TTD Target ID TTD Drug/Compound ID Pubchem CID Activity T34562 CANH78 17280 IC50 = 3270000 nM T34562 C27IRS 197934 IC50 = 1280000 nM T34562 CBJ36Y 639433 IC50 = 564130 nM T34562 CF2BD8 907361 IC50 = 21370 nM T34562 C5NQG3 940069 IC50 = 31410 nM T34562 CJGB43 941230 IC50 = 40000 nM T34562 CEX1K9 10243765 IC50 = 19050 nM T34562 C5I4SX 10402002 IC50 = 28980 nM T34562 C2JY8F 15388819 IC50 = 3000 nM T34562 C8G9AL 16756850 IC50 > 10000 nM T34562 C0SDW6 127025482 Ki = 2390 nM T34562 CK7L8U 127027355 IC50 = 23700 nM T34562 CH6ON2 127027684 IC50 = 625710 nM T34562 C7ST9X 127028306 IC50 = 317310 nM T34562 CN86IR 127028327 IC50 = 3333300 nM T34562 CHU16M 127028328 IC50 = 2064200 nM T34562 CV03TZ 127028660 IC50 = 237500 nM T34562 CBE6M2 127028661 IC50 = 627000 nM T34562 C5P3GA 127029548 IC50 = 8760 nM T34562 C1ZP4G 130431469 IC50 > 10000 nM T34562 CMA35H 130431481 IC50 > 10000 nM T34562 D0S9LT 12793 IC50 = 3250000 nM T34562 D0T0YI 378 IC50 = 18500000 nM T25464 D06OMK 445643 IC50 = 14.8 nM T25464 D0G7UX 5284373 IC50 = 183 nM T25464 C12CHL 4470793 Ki > 300000 nM T25464 C6YF5L 9918081 Ki > 3000 nM T25464 CC30ZA 10305301 Ki > 200000 nM T25464 C9TQ7U 11105029 IC50 = 2.8 nM T25464 C7WJF0 15546641 IC50 = 7.2 nM T25464 CU2A6K 44306123 IC50 = 7.32 nM T25464 C7WNM2 44306124 IC50 = 4.17 nM T25464 C86EOZ 44306135 IC50 = 8.65 nM T25464 C8T5NI 44306145 IC50 = 14 nM T25464 CUH17I 44306155 IC50 = 8.7 nM T25464 C6OQ4D 44306156 IC50 = 5.85 nM T25464 CN58YR 44306157 IC50 = 7.25 nM T25464 C8N7QZ 44306253 IC50 = 4.93 nM T25464 CD8O6N 44306280 IC50 = 7.91 nM T25464 C68IRQ 44306324 IC50 = 3.96 nM T25464 CBI4S6 44373943 IC50 > 5000 nM T25464 CQX6L4 44374010 IC50 = 348 nM T25464 C4I9DK 44374019 IC50 = 742 nM T25464 CBH09L 44374020 IC50 = 363 nM T25464 C89QDY 44374110 IC50 = 890 nM T25464 CQ65HS 44374127 IC50 > 5000 nM T25464 CJ9G7T 44374128 IC50 = 1539 nM T25464 C4XI8B 44374132 IC50 = 581 nM T25464 CYO20C 44374169 IC50 = 636 nM T25464 C1G6CI 44374400 IC50 = 840 nM T25464 CS30FH 49863381 IC50 = 140 nM T25464 C3YI2V 49863382 IC50 = 89 nM T25464 CS48JU 49863383 IC50 = 49 nM T71367 D0E3TC 44259 IC50 = 0.57 nM T71367 D00SDR 90054634 IC50 = 330 nM T71367 D0HK8C 90054733 IC50 = 121 nM T71367 D0L2FW 90054621 IC50 = 546 nM T71367 CA3C5S 3685259 IC50 < 5000 nM T71367 CACS26 11561968 Ki > 1000 nM T71367 CU0E8O 11690457 Ki > 1000 nM T71367 CJ21EH 13626914 IC50 = 94 nM T71367 C5VPH9 16129448 IC50 = 892 nM T71367 CGD89T 27126517 IC50 = 861 nM T71367 CC71QJ 27666048 IC50 > 100000 nM T71367 C61HBG 45102725 IC50 = 4200 nM T71367 CLS29B 46872626 IC50 > 10000 nM T71367 C5BZV3 57958821 IC50 = 381 nM T71367 C1MR8Q 60097495 IC50 > 1000 nM T71367 C37NKO 67129970 IC50 > 10000 nM T71367 CK80LJ 67130050 IC50 = 9430 nM T71367 CV63UL 67240318 IC50 > 10000 nM T71367 C7GRV2 68755406 IC50 > 10000 nM T71367 C7D2UQ 69463478 IC50 = 189 nM T71367 CVIA91 71553085 IC50 = 120 nM T71367 C1TR3O 71553152 IC50 = 2480 nM T71367 CDJY72 71568837 IC50 = 1600 nM T71367 C8CAG7 71578921 IC50 > 10000 nM T71367 C6P5YH 71657853 IC50 = 1.4 nM T71367 CKRS82 71678791 IC50 = 18 nM T71367 C7ROZ1 71679297 IC50 = 46 nM T71367 C9JTE7 71679299 IC50 = 16 nM T71367 C9RQW2 71679784 IC50 = 32 nM T71367 CHR3P5 71679785 IC50 = 15 nM T71367 CK1HR0 71679949 IC50 = 41 nM T71367 CF7R0Y 71682057 IC50 = 8000 nM T71367 CZM67T 72703518 IC50 = 150 nM T71367 C84AEF 72705109 IC50 = 77 nM T71367 CBK47T 72705487 IC50 = 132 nM T71367 CVF5P0 73603034 IC50 = 5700 nM T71367 C3SJQ2 76336279 IC50 > 100000 nM T71367 CI6NL9 77068235 IC50 = 8 nM T71367 C7RO1U 86703926 IC50 = 60 nM T71367 C97DVA 89729987 IC50 = 401 nM T71367 C2O4JR 89730033 IC50 = 3.5 nM T71367 C4UY2V 89730039 IC50 = 1.6 nM T71367 CB7Y0S 89730041 IC50 = 3.7 nM T71367 CQM98T 89730047 IC50 = 3.7 nM T71367 CC97QK 90054623 IC50 = 689 nM T71367 C93YPW 90054630 IC50 = 1700 nM T71367 CX0WH7 90054720 IC50 = 297 nM T71367 C9CRM6 90054726 IC50 = 423 nM T71367 CJX51L 90054730 IC50 = 225 nM T71367 CRF7M2 90054734 IC50 = 387 nM T71367 CEO7I0 90054986 IC50 = 58 nM T71367 CIZ2T6 90055028 IC50 = 351 nM T71367 C3ZV1C 90655985 IC50 = 5840 nM T71367 CE9KY0 90655986 IC50 = 2120 nM T71367 C6JIP7 91664348 IC50 = 4000 nM T71367 C18QYF 105539853 IC50 = 19.95 nM T71367 CBZ59D 118701008 IC50 = 3.7 nM T71367 C9CUL3 118711764 IC50 = 1600 nM T71367 CZH6E4 118711841 IC50 = 150 nM T71367 CYL46R 118711842 IC50 = 70 nM T71367 C2OK7E 118711843 IC50 = 710 nM T71367 CR8B9H 118711844 IC50 = 160 nM T71367 C5VDI0 118711845 IC50 = 840 nM T71367 C92TDH 118711846 IC50 = 300 nM T71367 C37IZJ 118711847 IC50 = 640 nM T71367 C8XFB1 118711848 IC50 = 130 nM T71367 COM51H 118711849 IC50 = 180 nM T71367 C7CB6W 118711850 IC50 = 10 nM T71367 CPNM74 118711851 IC50 = 70 nM T71367 C48DCS 118711852 IC50 = 10 nM T71367 CX8CL3 118711853 IC50 = 11000 nM T71367 CZV53F 118711854 IC50 = 19000 nM T71367 C2LT9G 118711855 IC50 = 37000 nM T71367 C0VBS5 118711856 IC50 = 7000 nM T71367 C0IJF5 118711857 IC50 = 23000 nM T71367 C7JV3C 118711858 IC50 = 3000 nM T71367 C4LJ6U 118711859 IC50 = 10000 nM T71367 C0QDO9 118711860 IC50 = 6000 nM T71367 CK0W1O 118711861 IC50 = 1000 nM T71367 C9XBL5 118711862 IC50 = 2000 nM T71367 CT3IS4 118711863 IC50 = 2000 nM T71367 C26EOM 118711864 IC50 = 1000 nM T71367 C9AGI1 118711865 IC50 = 2000 nM T71367 C2SQ6P 118711866 IC50 = 2000 nM T71367 C5GPJ9 118711891 IC50 = 2000 nM T71367 C76KYO 118711892 IC50 = 6000 nM T71367 CKBQ72 118711893 IC50 = 3000 nM T71367 CEU0S4 118711894 IC50 = 5000 nM T71367 CK63ES 118711895 IC50 = 10000 nM T71367 C92ZJE 118711896 IC50 = 8000 nM T71367 C2JA8B 127025153 IC50 = 600 nM T71367 CVUE54 127025154 IC50 = 84 nM T71367 C6W1UY 127025155 IC50 = 64 nM T71367 CLIP96 127026999 IC50 = 96 nM T71367 CEBO19 127027293 IC50 = 46 nM T71367 C5CUO0 127027294 IC50 = 248 nM T71367 CYS8L4 127027295 IC50 = 270 nM T71367 C39LPD 127027304 IC50 = 20 nM T71367 C3E7FZ 127028834 IC50 = 410 nM T71367 CJX04U 127029806 IC50 = 1509 nM T71367 CWVN31 127029807 IC50 = 1722 nM T71367 C9TZ7D 127034994 IC50 = 48 nM T71367 CE7M4J 127036775 IC50 = 14.9 nM T71367 CP89UZ 127036952 IC50 = 13 nM T71367 CX3Z7Q 134136970 IC50 > 100000 nM T71367 C82XFJ 134139661 IC50 > 100000 nM T71367 CKB1J9 134144378 IC50 = 44000 nM T71367 COF17E 134147249 IC50 = 5600 nM T71367 C60OFR 134154014 IC50 > 100000 nM T71367 CY4D8I 135566504 Ki = 812.4 nM T71367 CG3UZ1 135927974 Ki > 1000 nM T71367 CWGA76 137530158 IC50 = 12.59 nM T71367 CI1E8V 137634241 IC50 > 10000 nM T71367 C2E4DP 139592531 IC50 = 158.49 nM T71367 CZ7YS0 146027031 IC50 = 19.95 nM T71367 C2MD1Q 155513187 IC50 > 10000 nM T71367 CE7TI4 155521619 IC50 = 7943.28 nM T71367 CPW4H0 155531070 IC50 = 19952.62 nM T71367 CONB81 155557716 IC50 = 3981.07 nM T71367 D0NY6U 86703914 IC50 = 17 nM T71367 D0O6OH 71553154 IC50 = 18 nM T86928 D04AIT 5280445 IC50 = 500 nM T86928 D0K8KX 5280343 IC50 = 550 nM T86928 D0R3JB 4212 IC50 = 660 nM T86928 D09JEJ 24748573 IC50 = 3 nM T86928 D0B9BU 6918454 EC50 = 100 nM T86928 D0WS1V 448991 IC50 > 10000 nM T86928 C2OAV0 7328982 EC50 = 1600 nM T86928 CQVZ16 44123806 IC50 = 710 nM T86928 C1O6NR 44123807 IC50 = 480 nM T86928 C91MBN 44123808 IC50 = 820 nM T86928 CX08MT 44590715 IC50 = 2610 nM T86928 CVK4W9 44590746 IC50 = 2600 nM T86928 CO1UP9 44590747 IC50 = 5870 nM T86928 C3QRL8 44590749 IC50 = 2500 nM T86928 C4MY0L 44590794 IC50 = 8600 nM T86928 CLPU05 44590795 IC50 = 1520 nM T86928 C1CQS8 44590796 IC50 = 1100 nM T86928 C1MR8Q 60097495 IC50 > 10000 nM T86928 CPL8X0 139593287 EC50 = 6000 nM T86928 C7UNX2 145991479 IC50 < 1000 nM T86928 C2MD1Q 155513187 IC50 > 10000 nM T86928 C4PL1X 155536605 IC50 = 45100 nM T86928 CT9D0Q 155547691 IC50 = 18230 nM T86928 C2G8TU 155550182 IC50 = 1650 nM T86928 C1ACW9 155552233 IC50 = 8070 nM T86928 CDXK27 155562302 IC50 = 850 nM T86928 C6ICJ5 155562508 IC50 = 21990 nM T86928 CV74OB 155566389 IC50 = 4400 nM T86928 CGSU30 155566872 IC50 = 17750 nM T86928 D00RIX 5280443 IC50 = 800 nM T86928 D00YEV 5281605 IC50 = 10000 nM T86928 D01UYI 5281607 IC50 = 9000 nM T86928 D02DML 5281707 IC50 = 200 nM T86928 D07OAT 456214 IC50 > 10000 nM T86928 D0CP3M 5149739 IC50 = 930 nM T86928 D0G3TK 5280863 IC50 = 400 nM T86928 D0LH4L 10154 IC50 = 700 nM T86928 D0MF5Y 5281614 IC50 = 350 nM T86928 D0NJ4H 5281670 IC50 = 10000 nM T86928 D0O1YH 1694 IC50 = 1600 nM T86928 D0T3PW 5281672 IC50 = 900 nM T59102 D00STL 644241 IC50 = 71 nM T59102 D01PZD 5329098 IC50 = 68 nM T59102 D03ZBT 11626560 IC50 > 1000 nM T59102 D07POC 176870 IC50 = 12200 nM T59102 D08CDI 208908 IC50 = 8500 nM T59102 D09GDD 11167602 IC50 = 1.5 nM T59102 D09KTS 24821094 IC50 > 1000 nM T59102 D0AZ3C 5291 IC50 = 72 nM T59102 D0E6XR 3062316 Ki < 10 nM T59102 D0G6QF 3081361 IC50 = 1100 nM T59102 D0H0EQ 24826799 IC50 = 1.2 nM T59102 D0J9ZR 4477 IC50 > 100000 nM T59102 D0R0MW 5329102 IC50 = 2 nM T59102 D0W5HK 216239 IC50 = 37 nM T59102 D00UZR 5330286 IC50 > 10000 nM T59102 D02UFQ 11620908 IC50 > 10000 nM T59102 D03AND 11656518 IC50 = 6 nM T59102 D08HOM 46207586 IC50 = 3 nM T59102 D0A1AQ 5329099 IC50 = 50 nM T59102 D0D1GF 42642645 IC50 = 9.4 nM T59102 D0E3TC 44259 IC50 = 0.6 nM T59102 D0HS5V 11234052 IC50 > 6000 nM T59102 D0M0XB 10302451 IC50 > 5000 nM T59102 D0M9QZ 11485656 IC50 = 60 nM T59102 D0O0LS 25141092 IC50 > 10000 nM T59102 D0O6WV 24794418 IC50 > 500 nM T59102 D0P6DJ 151194 IC50 = 490 nM T59102 D0T2ER 24767976 IC50 = 13 nM T59102 D0Z6MT 16662431 IC50 = 4 nM T59102 D03BNU 59604787 IC50 > 3500 nM T59102 D0JY1I 42613483 IC50 = 3900 nM T59102 D06GBK 2048 IC50 = 6200 nM T59102 D0H4GI 10275001 IC50 = 406 nM T59102 D0IT6Q 3038522 IC50 = 26 nM T59102 D0L5YF 5329032 IC50 = 3400 nM T59102 D0T3ME 156422 IC50 = 6200 nM T59102 C63WLY 89644 IC50 > 10 ug.mL-1 T59102 C5JE2Z 104860 IC50 = 7.6 ug.mL-1 T59102 C6Y9CV 151193 IC50 = 490 nM T59102 CI1NA5 159926 IC50 > 10 ug.mL-1 T59102 CYBA43 177458 IC50 > 10 ug.mL-1 T59102 C32HFB 396514 IC50 = 2000 nM T59102 C4MNG8 445840 IC50 = 5000 nM T59102 C75EDQ 644355 IC50 = 100 nM T59102 C5HPF3 644356 IC50 = 20 nM T59102 C9D7UY 727518 IC50 > 100000 nM T59102 CXB5A2 964113 IC50 > 100000 nM T59102 CDB17F 1538822 IC50 = 24200 nM T59102 CZ2B4M 2358462 IC50 > 100000 nM T59102 CXA1L7 2365265 IC50 > 100000 nM T59102 CEF62M 2379240 IC50 = 33100 nM T59102 CKT64G 2396126 IC50 > 10000 nM T59102 CFVK40 3008950 IC50 > 50000 nM T59102 CD8UW1 3008956 IC50 = 17000 nM T59102 CCD93P 3008957 IC50 > 50000 nM T59102 CU64VM 3008958 IC50 > 50000 nM T59102 C8F0KM 3008959 IC50 > 50000 nM T59102 CV8R9Z 3008960 IC50 > 50000 nM T59102 C8EZ6O 3008961 IC50 > 50000 nM T59102 CX95SU 3008962 IC50 = 8900 nM T59102 C9B2MN 3008963 IC50 > 50000 nM T59102 C9E7BW 3008964 IC50 > 50000 nM T59102 CGK91Q 3008965 IC50 = 14700 nM T59102 CCN9D5 3142817 IC50 = 1000 nM T59102 CY28LS 5293755 IC50 > 100000 nM T59102 CFW19M 5329009 IC50 = 3000 nM T59102 C9I7WT 5329100 IC50 = 60 nM T59102 CMWB28 5329101 IC50 = 17 nM T59102 CGX50J 5329104 IC50 = 5 nM T59102 C2VX0H 5329105 IC50 = 0.5 nM T59102 CK71MQ 5329106 IC50 = 1 nM T59102 CL0Q4S 5329107 IC50 = 3 nM T59102 C6YRH8 5329108 IC50 = 2 nM T59102 CFP59Y 5329109 IC50 = 1 nM T59102 C0JW3Y 5329134 IC50 = 2110 nM T59102 CO7J2A 5329135 IC50 = 620 nM T59102 CQ4TP5 5329136 IC50 = 8290 nM T59102 CXQC42 5329137 IC50 = 11300 nM T59102 CT94JS 5329138 IC50 = 140 nM T59102 CNH06M 5329139 IC50 = 4190 nM T59102 CRY4Z2 5329140 IC50 = 5980 nM T59102 CAPE50 5329141 IC50 = 1400 nM T59102 CFU58A 5329142 IC50 = 160 nM T59102 C5Q8XK 5329143 IC50 = 170 nM T59102 C8PX4D 5329144 IC50 = 650 nM T59102 C6USQ5 5329145 IC50 = 2780 nM T59102 C56LWT 5329146 IC50 = 3650 nM T59102 CZ16MN 5329147 IC50 = 1210 nM T59102 CAN16I 5329148 IC50 = 1530 nM T59102 CG4NC2 5329149 IC50 = 550 nM T59102 CIW70H 5329150 IC50 = 110 nM T59102 C5FT6A 5329151 IC50 = 230 nM T59102 CB0N4L 5329152 IC50 = 940 nM T59102 COFP24 5329153 IC50 = 680 nM T59102 CGWD98 5329154 IC50 = 5460 nM T59102 C4PD0K 5329156 IC50 = 11500 nM T59102 C0RWT8 5329157 IC50 = 1030 nM T59102 C3MU5S 5329158 IC50 = 3460 nM T59102 CN6O4R 5329159 IC50 = 70600 nM T59102 CG68DI 5329160 IC50 > 100000 nM T59102 CYR7V0 5329161 IC50 = 13900 nM T59102 C9BXE2 5329162 IC50 = 94010 nM T59102 CY4V5Z 5329163 IC50 = 240 nM T59102 CI64YA 5329164 IC50 = 4 nM T59102 C2ZV0O 5329165 IC50 < 780 nM T59102 CAB53L 5329166 IC50 = 20 nM T59102 CTW9R8 5329167 IC50 = 19300 nM T59102 C8A3TJ 5329168 IC50 = 40 nM T59102 CVTD82 5329169 IC50 = 680 nM T59102 CQ5WK1 5329170 IC50 = 870 nM T59102 CNC9T7 5329171 IC50 = 5430 nM T59102 C6L0UW 5329229 IC50 > 20000 nM T59102 C1DBV6 5329230 IC50 > 20000 nM T59102 CLKM80 5329231 IC50 > 20000 nM T59102 CTQ18A 5329232 IC50 > 100000 nM T59102 CM5KG6 5329233 IC50 > 20000 nM T59102 CQG6R2 5329234 IC50 > 20000 nM T59102 CJ3A9I 5329235 IC50 > 100000 nM T59102 CPS7X1 5329236 IC50 > 100000 nM T59102 CAN60T 5329237 IC50 > 20000 nM T59102 CY15JP 5329238 IC50 > 20000 nM T59102 C41UBI 5329239 IC50 > 20000 nM T59102 C6VQ9F 5329240 IC50 > 20000 nM T59102 C8WS5K 5329241 IC50 > 20000 nM T59102 CI26UN 5329242 IC50 > 20000 nM T59102 C6PJ2R 5329243 IC50 > 20000 nM T59102 C0OKB7 5329244 IC50 = 20000 nM T59102 C78ZNL 5329245 IC50 > 20000 nM T59102 CWL5S4 5329246 IC50 = 20000 nM T59102 C4X3OE 5329248 IC50 = 5620 nM T59102 CK8FH6 5329249 IC50 > 20000 nM T59102 CN5B6C 5329250 IC50 > 20000 nM T59102 CQ0B6E 5329251 IC50 > 10000 nM T59102 C4KO3N 5329252 IC50 > 100000 nM T59102 C6MZF8 5329253 IC50 > 20000 nM T59102 C9NBG7 5330546 IC50 = 70 nM T59102 CS3A8F 5331081 IC50 > 20000 nM T59102 CG4W8K 5331082 IC50 > 20000 nM T59102 CD4C2A 5331083 IC50 > 20000 nM T59102 C6AT8V 5331084 IC50 > 20000 nM T59102 CJVS23 5331085 IC50 > 20000 nM T59102 CZ29FN 5331086 IC50 > 20000 nM T59102 CYL78A 5331087 IC50 > 20000 nM T59102 CJ87XR 5331088 IC50 = 2100 nM T59102 CFB3K7 5331089 IC50 = 18000 nM T59102 C9WY1O 5331090 IC50 > 20000 nM T59102 C9ZK3D 5331091 IC50 > 20000 nM T59102 C6RJC8 5331092 IC50 = 1100 nM T59102 C0IOY8 5331093 IC50 = 1400 nM T59102 CMD08O 5331094 IC50 = 1100 nM T59102 CDQ3M7 5359485 IC50 = 0.89 ug.mL-1 T59102 C54BYP 5360741 IC50 = 1.8 ug.mL-1 T59102 CD65JT 5427216 IC50 > 100000 nM T59102 CPB95V 5427224 IC50 > 100000 nM T59102 C61NCL 5482344 IC50 = 1800 nM T59102 CDK3J0 5703619 IC50 = 0.4 nM T59102 CA6L5V 5707304 IC50 > 100000 nM T59102 C43YGE 5713379 IC50 > 100000 nM T59102 CT8U7I 5874584 IC50 = 8390 nM T59102 CM8LW9 6036100 IC50 > 100000 nM T59102 C6L5HS 6419386 IC50 = 2800 nM T59102 C3CQW0 6419387 IC50 = 1000 nM T59102 CWOA63 6419388 IC50 = 2000 nM T59102 CZVU64 6419389 IC50 = 1400 nM T59102 C9FN4B 6419390 IC50 = 800 nM T59102 CN53YW 6419391 IC50 = 4000 nM T59102 C17NWJ 6419392 IC50 = 600 nM T59102 C13IRC 6419393 IC50 = 2000 nM T59102 C4FLE9 6419394 IC50 = 800 nM T59102 C4GHT0 6419395 IC50 = 4000 nM T59102 C8SAQ1 6419396 IC50 > 10000 nM T59102 CP71CL 6419397 IC50 > 10000 nM T59102 CQ3S8L 6450842 IC50 = 3700 nM T59102 C2N0IR 6477203 IC50 = 12800 nM T59102 CW5YJ2 6536705 IC50 > 100000 nM T59102 C2OL7K 9796455 IC50 = 353 nM T59102 CI80BK 9803350 IC50 = 2500 nM T59102 C9TAL6 9826308 IC50 = 160 nM T59102 CWVH12 9828619 IC50 = 50 nM T59102 CX10KR 9828962 IC50 = 170 nM T59102 CE5X8J 9844744 IC50 = 490 nM T59102 CSAY10 9845576 IC50 = 1500 nM T59102 C6A9HS 9871170 IC50 = 97 nM T59102 C3CI1J 9872659 IC50 = 20 nM T59102 CUZ07T 9884745 IC50 > 100000 nM T59102 CHF7G5 9890746 IC50 = 90 nM T59102 CXA5C8 9893493 IC50 > 2000 nM T59102 CZ25GL 9894619 IC50 = 70 nM T59102 C3EUB4 9911005 IC50 = 240 nM T59102 C24JTF 9911313 IC50 = 13300 nM T59102 C1Y3MH 9915808 IC50 = 90 nM T59102 C6HP3L 9948410 IC50 > 100000 nM T59102 C7T9DJ 9950440 IC50 > 30000 nM T59102 CO4N3Q 9995374 IC50 > 100000 nM T59102 C5WF7J 10007113 IC50 = 300 nM T59102 CY90DN 10023010 IC50 = 5 nM T59102 CJ95HR 10041745 IC50 = 12 nM T59102 CG57EC 10047098 IC50 = 13400 nM T59102 CUJR40 10062694 EC50 = 6 nM T59102 C1JUF8 10073832 IC50 > 2000 nM T59102 CIV15Q 10113978 IC50 = 84 nM T59102 C5WCL2 10117540 IC50 = 216 nM T59102 C5KHX2 10118413 IC50 = 50 nM T59102 C46DHW 10119600 IC50 = 230 nM T59102 CRNC72 10120038 IC50 = 90 nM T59102 C4VW8P 10121424 IC50 = 40 nM T59102 CYQ01B 10121530 IC50 = 30 nM T59102 CR5D2N 10121709 IC50 = 1 nM T59102 C5X7LQ 10121737 IC50 = 20 nM T59102 C3XW0Y 10122339 IC50 = 2.4 nM T59102 C6IA4L 10143909 IC50 = 77 nM T59102 C7X5LY 10145209 IC50 = 110 nM T59102 CL89XT 10165712 IC50 = 2 nM T59102 C76XOL 10166902 IC50 = 10 nM T59102 C1Y7HR 10167597 IC50 = 36 nM T59102 CR5Y7O 10168074 IC50 = 0.4 nM T59102 CJH54G 10186893 IC50 = 1430 nM T59102 C3ER4N 10187285 IC50 < 4 nM T59102 CM26BU 10187537 IC50 = 140 nM T59102 CA03YO 10187699 IC50 = 1010 nM T59102 CUG37L 10187829 IC50 = 335 nM T59102 C8T7RC 10188599 IC50 = 265 nM T59102 C6FB3Q 10188863 IC50 = 5040 nM T59102 C0N3HC 10189022 IC50 = 50 nM T59102 C6G2RK 10189131 IC50 = 20 nM T59102 CD4C9B 10207679 IC50 = 70 nM T59102 CZU79W 10208916 IC50 = 320 nM T59102 C4G2AD 10209993 IC50 = 9 nM T59102 CZJ78I 10210309 IC50 = 145 nM T59102 CBFZ09 10210632 IC50 = 99 nM T59102 C5YCN2 10215023 IC50 = 66000 nM T59102 C95ZXY 10226609 IC50 = 800 nM T59102 CB83CI 10228726 IC50 = 10 nM T59102 C18DRH 10229841 IC50 = 710 nM T59102 CD7J3O 10231458 IC50 = 20 nM T59102 CL9N2E 10231519 IC50 = 100 nM T59102 CAE03L 10231813 IC50 < 4 nM T59102 CPD6Z9 10236164 IC50 > 100000 nM T59102 CX15BI 10246728 IC50 = 3 nM T59102 C1WL8B 10251852 IC50 > 500000 nM T59102 CH30RC 10253133 IC50 = 1400 nM T59102 CBI47E 10264222 IC50 > 100000 nM T59102 C6DC8Q 10275163 IC50 = 3300 nM T59102 CD2IE3 10278606 IC50 = 920 nM T59102 CH5DQ0 10280082 IC50 = 140 nM T59102 C65JZS 10296462 IC50 = 1250 nM T59102 CVO54Z 10300451 IC50 > 20000 nM T59102 C63DPY 10301981 IC50 = 10 nM T59102 CO90LX 10302121 IC50 = 216 nM T59102 CC4G8B 10302519 IC50 < 4 nM T59102 C2T3WU 10302586 IC50 = 168 nM T59102 C4FP8M 10303591 IC50 < 4 nM T59102 C5CBF9 10320381 IC50 = 6600 nM T59102 C97YDQ 10344304 IC50 = 510 nM T59102 CZV0G7 10359698 IC50 = 16 nM T59102 CQB9H7 10389422 IC50 = 11000 nM T59102 CLAX64 10413508 IC50 = 11000 nM T59102 CQ43JU 10426229 IC50 = 17500 nM T59102 CU8JP3 10432698 IC50 = 1100 nM T59102 C95LYF 10457505 IC50 = 530 nM T59102 C7PLI5 10478569 IC50 > 2000 nM T59102 CJ5M1D 10482445 IC50 = 8000 nM T59102 CJWH60 10489322 IC50 > 100000 nM T59102 C5SVT4 10537949 IC50 > 100000 nM T59102 CGAW17 10562306 IC50 = 85400 nM T59102 C6AJI9 10562777 IC50 = 25500 nM T59102 CE5L6D 10587839 IC50 > 100000 nM T59102 CM8N6L 10593765 IC50 = 24500 nM T59102 CI30LZ 10613858 IC50 > 100000 nM T59102 CH6Z3L 10635478 IC50 = 65500 nM T59102 CB97UD 10636005 IC50 > 100000 nM T59102 C2UWA0 10658651 IC50 = 41700 nM T59102 C5L0IX 10663368 IC50 > 100000 nM T59102 C9Z7XH 10663503 IC50 = 49900 nM T59102 CH1G6P 10682457 IC50 > 100000 nM T59102 C54UAK 10728035 IC50 = 2800 nM T59102 CXSH91 10753550 IC50 = 18200 nM T59102 CVPW04 10755069 IC50 > 100000 nM T59102 C3WR0Q 10779668 IC50 > 100000 nM T59102 CF5T1H 10783444 IC50 > 100000 nM T59102 CX1DH7 10862508 IC50 = 6720 nM T59102 CU8P7M 10862866 IC50 = 2000 nM T59102 C54VTR 10863323 IC50 = 720 nM T59102 C43CLE 10863395 IC50 = 440 nM T59102 CD8M0L 10863993 IC50 = 8180 nM T59102 C71JKT 10873266 IC50 > 30000 nM T59102 C16FCD 10874104 IC50 = 18200 nM T59102 CY7E1M 10874618 IC50 = 160 nM T59102 CU92JA 10875187 IC50 = 1.4 nM T59102 CSTP13 10875630 IC50 = 26 nM T59102 C6QV1L 10885200 IC50 = 9420 nM T59102 C8TDN1 10885583 IC50 = 2210 nM T59102 C70PLZ 10885776 IC50 = 6500 nM T59102 CI4XR0 10885830 IC50 = 20 nM T59102 CRN57U 10895433 IC50 = 2570 nM T59102 CJSX79 10896366 IC50 = 4690 nM T59102 C0BN9J 10896386 IC50 = 150 nM T59102 CJ4P5T 10905857 IC50 = 850 nM T59102 CM5IA4 10906467 IC50 = 210 nM T59102 CO21NS 10907015 IC50 = 80 nM T59102 CB0MK5 10907225 IC50 = 150 nM T59102 C2IOU4 10907383 IC50 = 2810 nM T59102 CC3P6X 10907564 IC50 = 520 nM T59102 CJUI34 10917610 IC50 = 510 nM T59102 CCB49T 10917872 IC50 = 1040 nM T59102 C4WJ2T 10918068 IC50 = 715 nM T59102 C62LQW 10918358 IC50 = 290 nM T59102 C4OX0I 10918469 IC50 = 662 nM T59102 CS0BJ5 10928229 IC50 = 110 nM T59102 C1DS2G 10929540 IC50 = 440 nM T59102 C7MTO0 10929814 IC50 = 2970 nM T59102 CY0J9W 10951558 IC50 = 53 nM T59102 CJE7Y2 10961232 IC50 > 10000 nM T59102 C94GTN 10963029 IC50 = 5000 nM T59102 CBT4S3 10963044 IC50 = 29 nM T59102 CAC02X 10963192 IC50 = 500 nM T59102 CKD72X 10972606 IC50 = 9210 nM T59102 CL89QG 10973305 IC50 = 100 nM T59102 CPY51V 10983215 IC50 = 30 nM T59102 CCN5F8 10984279 IC50 = 3230 nM T59102 C9ELG2 10984685 IC50 = 222 nM T59102 CAP7E6 10995060 IC50 = 305 nM T59102 CB5AD7 11004892 IC50 = 230 nM T59102 C53QCD 11006148 IC50 = 177 nM T59102 C0LK2Q 11006502 IC50 = 494 nM T59102 CC87FE 11015336 IC50 = 1210 nM T59102 C71TOQ 11015640 IC50 > 30000 nM T59102 CY3B6O 11015880 IC50 = 330 nM T59102 C4F8ZN 11026804 IC50 > 30000 nM T59102 CDQ0H4 11027671 IC50 = 178 nM T59102 C59LQM 11027750 IC50 = 100 nM T59102 C4GLS2 11036639 IC50 = 11100 nM T59102 C9NYE2 11037955 IC50 = 290 nM T59102 CT5V2C 11039013 IC50 = 813 nM T59102 CL3FG7 11039428 IC50 = 0.4 nM T59102 CJ05CL 11048367 IC50 = 80 nM T59102 CWVC81 11049206 IC50 = 2310 nM T59102 C5V9DI 11049316 IC50 = 5590 nM T59102 CD9GY6 11049581 IC50 = 1260 nM T59102 C04QKG 11069972 IC50 = 2060 nM T59102 CXDA03 11070177 IC50 > 30000 nM T59102 CB7ND4 11071122 IC50 = 290 nM T59102 C0HM8T 11071223 IC50 = 160 nM T59102 CYG8V1 11071546 IC50 = 335 nM T59102 CV4R8X 11081103 IC50 = 740 nM T59102 CM04HI 11081393 IC50 = 60 nM T59102 CKX3Z5 11081446 IC50 = 220 nM T59102 C4G2AF 11091152 IC50 = 5360 nM T59102 CEB97L 11112669 IC50 = 1260 nM T59102 C4YUN5 11112927 IC50 > 30000 nM T59102 CQDC05 11113190 IC50 = 190 nM T59102 CYH21N 11113218 IC50 > 30000 nM T59102 CDZ80M 11114435 IC50 = 582 nM T59102 C5MAN7 11124388 IC50 = 300 nM T59102 C6HQ2L 11133954 IC50 = 480 nM T59102 CM9QT3 11143981 IC50 = 9960 nM T59102 C9KES6 11144730 IC50 = 790 nM T59102 CTJ9U3 11145086 IC50 = 1410 nM T59102 CU5DO2 11145515 IC50 = 20 nM T59102 C0D8CT 11155618 IC50 = 180 nM T59102 C7CNO9 11156466 IC50 = 100 nM T59102 CMJ31L 11156812 IC50 = 20 nM T59102 CBDS75 11157185 IC50 = 90 nM T59102 CP16ND 11168221 IC50 = 80 nM T59102 CL8Y4F 11177747 IC50 = 270 nM T59102 CWIT81 11178110 IC50 = 150 nM T59102 CCAG52 11179181 IC50 = 70 nM T59102 CK7B4X 11190431 IC50 > 30000 nM T59102 CBG94A 11191231 IC50 = 40 nM T59102 C7BHE0 11200526 IC50 = 4590 nM T59102 C09YIQ 11202821 IC50 > 30000 nM T59102 C65JPE 11212551 IC50 > 30000 nM T59102 C50JAG 11223943 IC50 = 1440 nM T59102 CN6BC7 11226164 IC50 > 30000 nM T59102 C87WCG 11226298 IC50 = 1390 nM T59102 CYA59I 11235645 IC50 > 30000 nM T59102 C0E1ML 11236566 IC50 = 140 nM T59102 C1QAS6 11237612 IC50 = 190 nM T59102 CH2VD7 11245435 IC50 > 30000 nM T59102 CGL6R0 11249274 IC50 = 200 nM T59102 CUV15L 11249319 IC50 > 30000 nM T59102 CKRA10 11258984 IC50 > 10000 nM T59102 C9F6KW 11260252 IC50 = 180 nM T59102 CC93YJ 11260253 IC50 > 30000 nM T59102 C6ZD4C 11270126 IC50 > 30000 nM T59102 CKI25P 11272815 IC50 = 70 nM T59102 CJW65Q 11273677 IC50 > 30000 nM T59102 C3IU8T 11281396 IC50 = 1300 nM T59102 C28XHQ 11282038 IC50 = 620 nM T59102 CZX0K9 11283270 IC50 = 550 nM T59102 C9I8AN 11293184 IC50 > 30000 nM T59102 C7I9TG 11293913 IC50 = 310 nM T59102 CIXK95 11295243 IC50 = 640 nM T59102 CYFT17 11295612 IC50 = 780 nM T59102 CNF7V4 11304951 IC50 > 30000 nM T59102 CVCE09 11305002 IC50 = 2700 nM T59102 CEN1J8 11306433 IC50 > 30000 nM T59102 C5PW1K 11306478 IC50 > 30000 nM T59102 CJ3N8G 11316908 IC50 > 30000 nM T59102 C41RWG 11318423 IC50 = 330 nM T59102 CVQ1Y0 11318736 IC50 = 20 nM T59102 C9G4YJ 11325945 IC50 > 30000 nM T59102 C2WKC3 11330812 IC50 > 30000 nM T59102 C15ZLJ 11340108 IC50 = 100 nM T59102 C4ICB0 11341503 IC50 = 650 nM T59102 C9K3LZ 11350308 IC50 = 1540 nM T59102 CV3K6Q 11351606 IC50 > 10000 nM T59102 C1LT5J 11352217 IC50 > 30000 nM T59102 CU18NY 11352407 IC50 = 3260 nM T59102 C24LHS 11353568 IC50 = 21000 nM T59102 C1UD0O 11372879 IC50 > 30000 nM T59102 CM4UY7 11373369 IC50 = 170 nM T59102 C25ZCN 11374110 IC50 = 130 nM T59102 C6EGP9 11374800 IC50 = 90 nM T59102 C8TLG4 11396174 IC50 = 380 nM T59102 CL19HT 11397589 IC50 = 810 nM T59102 C41NOY 11409644 IC50 = 80 nM T59102 CEG81P 11419763 IC50 = 130 nM T59102 C9IQP7 11419787 IC50 > 30000 nM T59102 C3NBZ9 11420151 IC50 = 6080 nM T59102 CMAI17 11420386 IC50 = 10200 nM T59102 CREQ51 11429654 IC50 = 96 nM T59102 CVQC06 11429694 IC50 > 30000 nM T59102 C9WEH6 11432198 IC50 = 60 nM T59102 C7AI2V 11432911 IC50 > 2000 nM T59102 C17WNX 11443611 IC50 = 90 nM T59102 C3SKT6 11443633 IC50 = 80 nM T59102 COF7Z1 11443718 IC50 > 30000 nM T59102 C6I2ER 11455034 IC50 = 100 nM T59102 CX5L2B 11464443 IC50 = 10300 nM T59102 CD3P4Q 11465678 IC50 = 390 nM T59102 CT34RJ 11466063 IC50 = 290 nM T59102 C6M9NC 11477626 IC50 > 2000 nM T59102 CEB29T 11490006 IC50 > 30000 nM T59102 C46JFZ 11494322 IC50 = 33 nM T59102 C9K8RE 11496022 IC50 = 137 nM T59102 CY72AM 11496228 IC50 = 659 nM T59102 C5UEK0 11510816 IC50 = 110 nM T59102 CG3BZ9 11517980 IC50 = 4 nM T59102 CFQ42U 11525980 IC50 = 23 nM T59102 CL7X4Q 11530963 IC50 = 1867 nM T59102 CID2P7 11536421 IC50 = 54 nM T59102 C6IOJ4 11546085 IC50 = 310 nM T59102 CF28TK 11565353 IC50 = 217 nM T59102 CZ1H0X 11569258 IC50 = 5500 nM T59102 CRL95F 11569396 IC50 = 1 nM T59102 CO9KP5 11583459 IC50 > 10000 nM T59102 CB91RQ 11589811 IC50 = 40 nM T59102 CM65QP 11590120 IC50 = 3 nM T59102 C69FYK 11604142 Ki = 200 nM T59102 CEG5W8 11608830 IC50 = 9 nM T59102 C8IKG5 11616255 IC50 = 458 nM T59102 CCB3X0 11617740 IC50 = 6220 nM T59102 CSM62L 11626920 IC50 = 31 nM T59102 CK34LS 11632737 IC50 = 200 nM T59102 C7W3TE 11633427 IC50 = 10 nM T59102 C5R6DG 11634086 IC50 > 800 nM T59102 C8V0YT 11639969 IC50 = 1200 nM T59102 CZM9K1 11675974 IC50 = 410 nM T59102 C3M1CF 11682291 IC50 = 5420 nM T59102 CCX2F5 11682611 IC50 = 0.4 nM T59102 C8AEX7 11687971 IC50 = 151900 nM T59102 CHG14R 11688408 IC50 = 55 nM T59102 CZY05V 11719421 IC50 = 6 nM T59102 CUB2N6 11719537 IC50 = 5 nM T59102 C9P0VD 11729539 IC50 = 550 nM T59102 CBL38T 11730367 IC50 = 260 nM T59102 C4PE0D 11730369 IC50 = 1140 nM T59102 C3DVE0 11730809 IC50 = 370 nM T59102 CCQO28 11731042 IC50 = 871 nM T59102 C23STH 11731130 IC50 = 601 nM T59102 CSLC27 11731197 IC50 = 50 nM T59102 C5NLG6 11732326 IC50 = 3180 nM T59102 CU54IA 11732691 IC50 > 30000 nM T59102 C2M7ZD 11733137 IC50 = 1240 nM T59102 C67FZJ 11734285 IC50 = 400 nM T59102 CT49LJ 11734851 IC50 = 12 nM T59102 CU9BR4 11749848 IC50 > 30000 nM T59102 C0QV3M 11752083 IC50 = 10900 nM T59102 CAS0V7 11752632 IC50 = 290 nM T59102 CP7AH3 11755812 IC50 = 7700 nM T59102 CRW2H3 11762328 IC50 = 21600 nM T59102 CRI64Z 11762329 IC50 = 1200 nM T59102 CJI7T6 11763085 IC50 = 76 nM T59102 C61QXW 11785508 IC50 > 30000 nM T59102 CEOH20 11813259 IC50 = 943 nM T59102 C89SNG 11813434 IC50 > 30000 nM T59102 C4V8PJ 11813761 IC50 = 110 nM T59102 C1CI6M 11826385 IC50 = 440 nM T59102 CEUB71 11826832 IC50 = 1470 nM T59102 C9EV8H 11827121 IC50 = 3110 nM T59102 C72RZN 11827714 IC50 = 720 nM T59102 C14MZC 11827841 IC50 = 6750 nM T59102 CDZ1I3 11989153 IC50 = 637 nM T59102 CM50UH 12000646 EC50 = 170 nM T59102 CI39TK 12004372 IC50 = 10700 nM T59102 CDGF78 15282555 IC50 = 3300 nM T59102 C7LB4I 15949613 IC50 = 96 nM T59102 C9TU1O 16046126 IC50 > 1000 nM T59102 CW2XK6 16050925 IC50 = 110 nM T59102 C9JK2M 16059071 IC50 > 2000 nM T59102 CW6UJ9 16059338 IC50 > 1000 nM T59102 CH7MS6 16059729 IC50 > 42000 nM T59102 CFKE48 16064750 IC50 = 1 nM T59102 CQG45C 16109001 IC50 = 1940 nM T59102 C5VPH9 16129448 IC50 = 5270 nM T59102 C0V8FB 16730091 IC50 = 2 nM T59102 CA24TE 16730092 IC50 = 5 nM T59102 CGX61W 22041319 IC50 = 10 nM T59102 CYP32E 22707343 IC50 = 540 nM T59102 CFO6J5 22707344 IC50 = 10700 nM T59102 CWXO86 22707354 IC50 = 1320 nM T59102 C8JD2X 22707384 IC50 > 750 nM T59102 CAG61Z 22707433 IC50 = 2880 nM T59102 C20RYA 22707442 IC50 = 1380 nM T59102 CNR0O7 22707450 IC50 = 5160 nM T59102 CEOV57 22707452 IC50 > 100 nM T59102 CPO51J 22707462 IC50 = 6250 nM T59102 CGR94W 22707466 IC50 = 500 nM T59102 C3H1VE 22707498 IC50 = 1160 nM T59102 CDI35F 22707517 IC50 > 30000 nM T59102 C6MBW9 22707526 IC50 = 970 nM T59102 CQ3TW0 22707568 IC50 = 29700 nM T59102 CB29GC 22707603 IC50 = 350 nM T59102 C2UO3S 22707619 IC50 > 30000 nM T59102 CM5R8B 22707669 IC50 = 1120 nM T59102 C7G6NJ 22707741 IC50 = 5170 nM T59102 C9QLP0 23133323 IC50 = 1100 nM T59102 CG12OL 23518511 IC50 > 20000 nM T59102 CRX0Q6 23625758 IC50 = 780 nM T59102 C2RV3U 24180608 IC50 > 30000 nM T59102 C3X1WH 24742411 IC50 = 2 nM T59102 CS78XJ 24742412 IC50 = 3 nM T59102 C2KA6G 24742584 IC50 = 4 nM T59102 CN9GC8 24742586 IC50 = 10 nM T59102 CHU49V 24757938 IC50 < 1 nM T59102 C0D2PA 24758868 IC50 = 20 nM T59102 C3K5YO 24758982 IC50 = 7 nM T59102 CYU0Z8 24758983 IC50 = 6 nM T59102 CJL67N 24759089 IC50 = 4 nM T59102 C2APK8 24759090 IC50 = 9 nM T59102 C5CRF6 24759091 IC50 = 6 nM T59102 CA8U7X 24759094 IC50 = 4 nM T59102 CRB89L 24759205 IC50 = 1 nM T59102 C13JUP 24759314 IC50 = 5 nM T59102 CCPS81 24764502 IC50 > 35000 nM T59102 C9B2TF 24880043 IC50 = 150 nM T59102 CFK2B9 24882503 IC50 = 1400 nM T59102 C43HWQ 24883287 IC50 > 10000 nM T59102 C8DA5Q 24883334 IC50 > 10000 nM T59102 C4V9GH 24894117 IC50 = 11000 nM T59102 CJH19T 24894883 IC50 = 45000 nM T59102 CB5TP8 24894992 IC50 = 38000 nM T59102 CF4N9X 24895100 IC50 = 40000 nM T59102 CY8L7E 24896769 IC50 > 10000 nM T59102 CN13JF 24899915 IC50 = 1.3 ug.mL-1 T59102 CBWR97 24899916 IC50 = 1.8 ug.mL-1 T59102 C9F2JD 24899917 IC50 > 10 ug.mL-1 T59102 C64MTI 24900160 IC50 = 5.8 ug.mL-1 T59102 CO2I6Q 24900161 IC50 > 10 ug.mL-1 T59102 C5FD1A 24937369 IC50 = 5300 nM T59102 C4KG0Y 25022599 IC50 > 1000 nM T59102 CRO0Y8 25022735 IC50 = 90000 nM T59102 C72AJM 25022736 IC50 > 500000 nM T59102 CQ27UI 25113814 IC50 = 10 nM T59102 C2IHY0 25114266 IC50 = 5 nM T59102 CP8S9W 25116064 IC50 = 11 nM T59102 CTV54O 25123227 IC50 = 14 nM T59102 C1IYN7 25127854 IC50 = 5.9 nM T59102 CKD14B 25127856 IC50 = 19 nM T59102 CJBX60 25128180 IC50 = 8.3 nM T59102 CC5SD9 25128181 IC50 = 21 nM T59102 CIG4H0 25178539 IC50 = 4200 nM T59102 C4GI6J 25178540 IC50 = 6700 nM T59102 CL0Z1F 25181502 IC50 = 830 nM T59102 COB9G8 25181586 IC50 = 2800 nM T59102 C8YLD6 25194331 IC50 = 5 nM T59102 CXC9B3 25194865 IC50 = 9 nM T59102 C1I0VS 25194866 IC50 = 3 nM T59102 C9OZN3 25194867 IC50 = 30 nM T59102 C6FGQ1 25206346 IC50 = 91 nM T59102 CXNW87 25207322 IC50 = 8 nM T59102 C8IJB9 25218207 IC50 = 40300 nM T59102 C2TXC6 25218656 IC50 > 2000 nM T59102 CVM13K 42596931 IC50 = 100 nM T59102 CU53WB 42596953 IC50 = 2500 nM T59102 C7GIQ3 42625508 IC50 = 4600 nM T59102 CVZ83M 42625582 IC50 = 2700 nM T59102 C5MD9E 42625892 IC50 = 7300 nM T59102 CJ5U1X 42639664 IC50 = 6.4 ug.mL-1 T59102 CEL61X 44229839 IC50 > 10000 nM T59102 C4NWP5 44246325 IC50 > 200000 nM T59102 C2EW0I 44246326 IC50 = 118000 nM T59102 CSD8T0 44246327 IC50 > 200000 nM T59102 CMKF08 44246328 IC50 > 200000 nM T59102 CAO87V 44246329 IC50 > 200000 nM T59102 CLU2V3 44246330 IC50 = 17400 nM T59102 CHZ6Q1 44269004 IC50 = 10 nM T59102 CY6WC0 44299236 IC50 = 13000 nM T59102 C3RG0C 44299304 IC50 = 2300 nM T59102 CJM26I 44299321 IC50 = 4700 nM T59102 C9UGL3 44299325 IC50 = 10000 nM T59102 CJEZ96 44299338 IC50 = 9000 nM T59102 C8XGN5 44299339 IC50 = 5100 nM T59102 CNH34G 44299354 IC50 = 5600 nM T59102 C82MSD 44299360 IC50 = 18000 nM T59102 CSY8A3 44321301 IC50 > 100000 nM T59102 CCG2M5 44321317 IC50 = 60400 nM T59102 CY9ED1 44321395 IC50 > 100000 nM T59102 C5U1CR 44321686 IC50 > 10000 nM T59102 CETY53 44321717 IC50 = 66000 nM T59102 CV60ME 44321734 IC50 = 13800 nM T59102 C61OFE 44332377 IC50 > 1000 nM T59102 CI2NP3 44332378 IC50 = 160 nM T59102 CHKA01 44332616 IC50 = 820 nM T59102 CYAU21 44349046 IC50 = 409 nM T59102 CWFI13 44349291 IC50 = 564 nM T59102 C18OEK 44349292 IC50 = 50 nM T59102 C8XZ0Q 44349293 IC50 = 292 nM T59102 CYV2D7 44368815 IC50 = 357 nM T59102 CG6NE0 44394479 IC50 = 450 nM T59102 C6QL8A 44394480 IC50 = 970 nM T59102 C1BQ6T 44394484 IC50 = 240 nM T59102 CZ10CS 44394568 IC50 = 3590 nM T59102 CUF85K 44394571 IC50 = 400 nM T59102 CHO52Q 44394593 IC50 = 1010 nM T59102 CHCY97 44394612 IC50 = 2930 nM T59102 C7AB5H 44394617 IC50 = 350 nM T59102 C8M2PH 44394619 IC50 = 90 nM T59102 C58FRU 44394632 IC50 = 460 nM T59102 CB5S0R 44394633 IC50 = 220 nM T59102 CGLU71 44394634 IC50 = 10 nM T59102 CDU4J7 44394635 IC50 = 10 nM T59102 C4ZS5C 44394664 IC50 = 1150 nM T59102 C4ADU7 44394665 IC50 = 1400 nM T59102 C79BHS 44394670 IC50 = 180 nM T59102 CM0GF2 44394673 IC50 = 920 nM T59102 CF31RW 44394679 IC50 = 5 nM T59102 C53PUJ 44394680 IC50 = 280 nM T59102 C2JT4Q 44394704 IC50 = 770 nM T59102 C15GEC 44394709 IC50 = 1060 nM T59102 C6AEU0 44394722 IC50 = 5 nM T59102 C1GNQ7 44394737 IC50 = 4090 nM T59102 C2OAX3 44394745 IC50 = 510 nM T59102 C9RBN1 44394760 IC50 = 20 nM T59102 C6SRC1 44394772 IC50 = 1540 nM T59102 C70JWY 44394773 IC50 = 430 nM T59102 CPT6I0 44394781 IC50 = 3760 nM T59102 CLDS93 44394803 IC50 = 420 nM T59102 C81CTG 44394822 IC50 = 70 nM T59102 CRA0U1 44394842 IC50 = 2000 nM T59102 C0O8HG 44394845 IC50 = 630 nM T59102 C5PD3W 44394846 IC50 = 3090 nM T59102 C97CVT 44394847 IC50 = 100 nM T59102 CLT7U8 44394848 IC50 = 550 nM T59102 CD4U9G 44394849 IC50 = 590 nM T59102 CH8D0U 44394850 IC50 = 3420 nM T59102 CGOD34 44394853 IC50 = 2370 nM T59102 C6QNI1 44394865 IC50 = 80 nM T59102 CE8HO9 44394869 IC50 = 60 nM T59102 C43HND 44394870 IC50 = 100 nM T59102 C1L0SE 44394874 IC50 = 31700 nM T59102 CSE64J 44394875 IC50 = 370 nM T59102 C0XSD5 44394876 IC50 = 800 nM T59102 CW1QA3 44394898 IC50 = 13400 nM T59102 CFC1S9 44394899 IC50 = 160 nM T59102 C6GFO1 44394903 IC50 = 2130 nM T59102 CARP42 44394904 IC50 = 5190 nM T59102 CCT0R3 44394905 IC50 = 100 nM T59102 C8VJ2E 44405089 IC50 = 17 nM T59102 C8K4AL 44407237 IC50 > 50000 nM T59102 CUA18B 44407238 IC50 = 7600 nM T59102 C04HFE 44407248 IC50 > 50000 nM T59102 CR3O1C 44407275 IC50 = 15900 nM T59102 C70BFV 44407276 IC50 = 10200 nM T59102 CMH7W6 44407277 IC50 = 8700 nM T59102 C8W5YG 44447872 IC50 = 6 nM T59102 CUB12D 44449577 IC50 = 389 nM T59102 C3ZBV8 44450546 IC50 = 920 nM T59102 CLK0W7 44453682 IC50 > 1000 nM T59102 C0LY6E 44552561 IC50 = 6100 nM T59102 C7KRU3 44552562 EC50 = 2000 nM T59102 CYV71I 44555430 IC50 = 12.3 nM T59102 CJ1X9V 44565013 IC50 > 10000 nM T59102 CN2Q3D 44565014 IC50 = 1100 nM T59102 CM2GN3 44565015 IC50 > 10000 nM T59102 CV91YE 44572385 IC50 = 2600 nM T59102 C3CB2K 44572429 IC50 = 7800 nM T59102 CM2Q8J 44572430 IC50 = 5200 nM T59102 CAN4B0 44572431 IC50 = 1100 nM T59102 CMAT21 44572489 IC50 = 71000 nM T59102 CU1SY9 44572490 IC50 = 8700 nM T59102 CSD74G 44572491 IC50 = 13000 nM T59102 CA9WO3 44572537 IC50 = 47000 nM T59102 C06SLW 44572538 IC50 = 28000 nM T59102 CY8TG3 44572539 IC50 = 11000 nM T59102 C1JR4C 44572540 IC50 = 40000 nM T59102 CZ0PA9 44572581 IC50 = 2100 nM T59102 CD9VR5 44572582 IC50 = 13000 nM T59102 CG5UK0 44572584 IC50 = 11000 nM T59102 CMX32U 44572633 IC50 = 6200 nM T59102 C5WOE2 44586449 IC50 = 11800 nM T59102 C0VF8M 44586450 IC50 > 50000 nM T59102 C4K7NP 44586451 IC50 > 50000 nM T59102 C1JNR5 44586452 IC50 = 13700 nM T59102 C6T8UP 44586490 IC50 > 500000 nM T59102 CU95NI 44586526 IC50 = 100400 nM T59102 CBK9R3 44586527 IC50 > 500000 nM T59102 CA18IW 44586528 IC50 > 500000 nM T59102 C0YSZ2 44586577 IC50 = 77400 nM T59102 C8M5KI 44611919 IC50 = 22.8 nM T59102 C4KWJ3 45379956 IC50 > 50000 nM T59102 C2CU0B 45380067 IC50 > 50000 nM T59102 C6E2SC 45482700 IC50 > 10000 nM T59102 CZXH74 45482750 IC50 > 10000 nM T59102 CNI92D 46182735 IC50 = 230 nM T59102 CUA97D 46209401 IC50 = 120 nM T59102 C8YPN0 46225596 IC50 > 10000 nM T59102 C34JTS 46225597 IC50 = 5100 nM T59102 CGD73B 46225598 IC50 = 9100 nM T59102 C3E0PU 46225599 IC50 = 10000 nM T59102 CRDY89 46225610 IC50 = 3600 nM T59102 C0JMT8 46225611 IC50 > 10000 nM T59102 CF0D5J 46225612 IC50 = 1400 nM T59102 CFVO38 46225632 IC50 = 8700 nM T59102 CLZ1O6 46225634 IC50 = 4400 nM T59102 C07VDX 46225635 IC50 = 3800 nM T59102 CT70DX 46225640 IC50 = 7900 nM T59102 CJUF68 46225641 IC50 = 7700 nM T59102 C6AJ5N 46225647 IC50 = 3400 nM T59102 C2WCV1 46225648 IC50 = 9900 nM T59102 CBS96A 46225649 IC50 > 10000 nM T59102 C38BFC 46225657 IC50 = 2100 nM T59102 CD0A6F 46225658 IC50 > 10000 nM T59102 C1B3KS 46225663 IC50 = 2100 nM T59102 CU46XI 46225664 IC50 = 8000 nM T59102 CO3HS2 46225665 IC50 > 10000 nM T59102 C2UV1S 46225666 IC50 = 8200 nM T59102 CX5B1G 46225667 IC50 = 9200 nM T59102 C2Q9OH 46225668 IC50 > 10000 nM T59102 CM14FH 46225680 IC50 > 10000 nM T59102 CQS96E 46225681 IC50 > 10000 nM T59102 CJIK35 46225682 IC50 = 3800 nM T59102 C8S4QA 46225688 IC50 = 6700 nM T59102 C2P9QO 46228508 IC50 = 1550 nM T59102 C6E5PY 46228822 IC50 = 7490 nM T59102 C3T8AM 46228951 IC50 = 2390 nM T59102 CYZV41 46231219 IC50 = 2667 nM T59102 C7J5UP 46231220 IC50 = 858 nM T59102 CC96GZ 46231221 IC50 = 900 nM T59102 C9H4YO 46233889 IC50 = 49 nM T59102 CRT34L 46235770 IC50 = 27 nM T59102 CFR1C6 46845026 IC50 > 300000 nM T59102 C7NUY3 46847552 IC50 > 1000 nM T59102 CE3WH9 46865125 IC50 > 200000 nM T59102 C45LYT 46865445 IC50 > 200000 nM T59102 C1XEY4 46866615 IC50 > 200000 nM T59102 CF6K3E 46866616 IC50 > 200000 nM T59102 CA57MX 46886970 IC50 = 24600 nM T59102 CRGH62 46886971 IC50 = 183100 nM T59102 C68AGR 46886972 IC50 > 300000 nM T59102 CP32GW 46886973 IC50 > 300000 nM T59102 C48JWD 46886974 IC50 > 300000 nM T59102 C7H3MD 46887038 IC50 = 174900 nM T59102 C40NOR 46887039 IC50 = 43000 nM T59102 C7I4SB 46887074 IC50 = 182000 nM T59102 CI5QX2 46887110 IC50 = 171300 nM T59102 C0Q7NG 46887111 IC50 = 220400 nM T59102 CU15AN 46887112 IC50 = 110100 nM T59102 CD90BV 46887113 IC50 = 142200 nM T59102 CH3O9K 46887255 IC50 = 8500 nM T59102 C7NUT3 46887298 IC50 > 500000 nM T59102 CWV65D 46887299 IC50 > 500000 nM T59102 CH5BZ6 46887300 IC50 = 192400 nM T59102 C20UCB 46887348 IC50 > 500000 nM T59102 C0KEG5 46887349 IC50 > 500000 nM T59102 CY59RB 46887397 IC50 = 104200 nM T59102 C0WYM1 46898022 IC50 = 10000 nM T59102 CB92VU 46912443 IC50 = 2800 nM T59102 CU6HC7 46912444 IC50 = 34800 nM T59102 C8A4KU 46912445 IC50 > 500000 nM T59102 CNOS56 46912446 IC50 = 1300 nM T59102 CV38NE 46912546 IC50 > 500000 nM T59102 CQLT07 46913878 IC50 < 1000 nM T59102 CHSF07 49806372 IC50 > 1000 nM T59102 CVS85M 49831162 IC50 = 58 nM T59102 CR58WT 49840391 IC50 = 3 nM T59102 CA2J6U 49840467 IC50 = 13 nM T59102 CB0S2P 49842666 IC50 = 9200 nM T59102 C0NA9U 49842670 IC50 > 100000 nM T59102 CAI20B 49842778 IC50 = 21000 nM T59102 CRA74I 49842779 IC50 = 42000 nM T59102 CF91RS 49843531 IC50 > 10000 nM T59102 CE7D2J 49855568 IC50 = 3300 nM T59102 CFD9P3 49855569 IC50 = 1100 nM T59102 C1AU5N 49855758 IC50 = 2300 nM T59102 CIFK93 49855759 IC50 = 4000 nM T59102 CK48OJ 49855760 IC50 = 2300 nM T59102 CZI3M1 49855761 IC50 = 3900 nM T59102 CRPZ58 49855949 IC50 = 2500 nM T59102 CTU0K3 49855950 IC50 = 2700 nM T59102 CF85NL 49855951 IC50 = 4700 nM T59102 CF7YS9 49855952 IC50 = 1000 nM T59102 CJU38G 49855953 IC50 = 1800 nM T59102 CD2K4R 50908681 Ki > 1000000 nM T59102 C2Y6QS 50938552 IC50 > 10000 nM T59102 C9NYP4 51036677 IC50 > 10000 nM T59102 C4WRY3 51037112 IC50 > 10000 nM T59102 CRI28Z 51037948 IC50 > 10000 nM T59102 C4R7IM 52941368 IC50 = 71700 nM T59102 C7BY6M 52942956 IC50 > 200000 nM T59102 CA62KU 52944152 IC50 = 88200 nM T59102 CQV34K 52945403 IC50 > 200000 nM T59102 C97XZA 52946619 IC50 > 200000 nM T59102 CE0X5U 52947574 IC50 = 348000 nM T59102 CD9S4I 52947801 IC50 > 200000 nM T59102 CA6IL3 52947802 IC50 > 200000 nM T59102 C2KAJ4 52948634 IC50 > 500000 nM T59102 C0A1GQ 52949915 IC50 > 500000 nM T59102 C09SDH 53257410 IC50 > 10000 nM T59102 CZY0J7 53323592 IC50 > 100000 nM T59102 CNPM14 53341082 IC50 > 3000 nM T59102 C0SWH5 53348216 IC50 > 40000 nM T59102 CBK9Q6 53357848 IC50 > 10000 nM T59102 C8NA4L 53384644 IC50 > 30000 nM T59102 CVG90B 53389651 IC50 > 10000 nM T59102 C0JMY7 54673975 IC50 = 50500 nM T59102 C8AB1J 54759606 Ki = 19 nM T59102 CQ17GA 56640518 IC50 > 200000 nM T59102 CG20VK 56640520 IC50 > 200000 nM T59102 CZ9C8M 56640588 IC50 > 200000 nM T59102 CH0D7P 56640590 IC50 > 200000 nM T59102 C9DX3J 56649281 IC50 = 26 nM T59102 CR50TJ 56835147 IC50 = 2788 nM T59102 CI5ZJ7 56835161 IC50 > 100000 nM T59102 C2ML5S 56837168 IC50 = 518 nM T59102 CCW89V 56932477 IC50 = 185 nM T59102 CR3FK5 56932525 IC50 = 8 nM T59102 CY36EG 56945171 IC50 = 49 nM T59102 C4OG7H 56945172 IC50 = 93 nM T59102 CH0QA3 56945173 IC50 = 190 nM T59102 CM0NQ5 56945174 IC50 = 1100 nM T59102 CXKF03 56945175 IC50 = 550 nM T59102 CE07AQ 56945176 IC50 = 1600 nM T59102 CU86KC 56945272 IC50 = 23 nM T59102 C9SX7F 56945273 IC50 = 27 nM T59102 CG7VH5 56945274 IC50 = 72 nM T59102 C6WU4V 56945277 IC50 = 19 nM T59102 C7U9SL 56951304 IC50 > 50000 nM T59102 C0GQ9I 56951305 IC50 > 300000 nM T59102 C5YT6A 56951306 IC50 = 8920 nM T59102 CB03EH 56951307 IC50 = 193200 nM T59102 CP58NG 56954518 IC50 = 5 nM T59102 CAK91L 56955954 IC50 > 3600 nM T59102 C4YFJ5 57384105 IC50 = 1500 nM T59102 CV9RW5 57384106 IC50 = 1800 nM T59102 C4WE9B 57391179 IC50 = 10 nM T59102 CY10TP 57391180 IC50 = 6 nM T59102 CR4T2Y 57391283 IC50 = 129100 nM T59102 CU3DM9 57391295 IC50 > 1000 nM T59102 CBL74E 57392425 IC50 = 44300 nM T59102 CU7J9C 57393063 IC50 = 2 nM T59102 CD4HS3 57393074 IC50 = 9 nM T59102 CS60KL 57393075 IC50 > 2000 nM T59102 CWMT98 57394785 IC50 > 1000 nM T59102 CG18LI 57394786 IC50 = 34200 nM T59102 CEDP89 57394787 IC50 = 129300 nM T59102 C9PY4Q 57394798 IC50 = 10 nM T59102 C3F9VS 57394799 IC50 = 700 nM T59102 CP6W4C 57394879 IC50 > 500000 nM T59102 CVR13L 57394880 IC50 > 500000 nM T59102 CA4Q3Y 57395925 IC50 = 145900 nM T59102 C4CN6V 57396453 IC50 = 10 nM T59102 CCT58R 57396454 IC50 > 200 nM T59102 CXA5Z9 57396541 IC50 = 2 nM T59102 CPAH35 57396542 IC50 = 4 nM T59102 CUGP85 57396545 IC50 = 212400 nM T59102 CY8U1Q 57396557 IC50 = 0.9 nM T59102 CBUP96 57396646 IC50 = 159600 nM T59102 CWV96N 57398329 IC50 = 3 nM T59102 C8K1WJ 57398330 IC50 = 0.3 nM T59102 CXJ68F 57398331 IC50 = 229600 nM T59102 CBK02S 57399984 IC50 = 1 nM T59102 CNU4I7 57399985 IC50 = 2 nM T59102 CD9KF3 57399986 IC50 = 2 nM T59102 C0BA7P 57401686 IC50 = 20 nM T59102 CH56JP 57401785 IC50 = 3 nM T59102 C7YMG1 57401804 IC50 = 300 nM T59102 C20ZAX 57401805 IC50 = 4 nM T59102 C15YQW 57401806 IC50 = 20 nM T59102 CY5TJ9 57401807 IC50 = 4 nM T59102 C4L0SA 57401808 IC50 = 0.4 nM T59102 C4J0OD 57403506 IC50 = 0.8 nM T59102 CN0M3Z 57403518 IC50 = 300 nM T59102 CZSM95 57412684 IC50 > 10000 nM T59102 CN53XW 57428969 IC50 = 57.3 nM T59102 CE59QS 57505507 IC50 = 5.5 nM T59102 C8P6RD 57505528 IC50 = 15 nM T59102 C8R4FE 57991377 IC50 = 125.4 nM T59102 CH7L5N 58172700 IC50 = 768.4 nM T59102 C4V7FY 58191950 IC50 = 16000 nM T59102 CPCA29 58191961 IC50 = 70000 nM T59102 C7HF1L 58191965 IC50 = 7200 nM T59102 C8LWY9 58191997 IC50 = 28000 nM T59102 C4IBV1 59375998 IC50 = 12.7 nM T59102 CV8Q2D 59376002 IC50 = 89.9 nM T59102 CL3ND8 59376009 IC50 = 7.6 nM T59102 CC2AF9 59376012 IC50 = 19.4 nM T59102 CR7CG3 59376014 IC50 = 22.7 nM T59102 C60RIS 59376021 IC50 = 41.6 nM T59102 CT3Q5G 59376025 IC50 = 21.3 nM T59102 C97YSI 59376026 IC50 = 64.8 nM T59102 CEH5X6 59376027 IC50 = 40.1 nM T59102 C79EBT 59376032 IC50 = 40.7 nM T59102 C06DNI 59376037 IC50 = 12.1 nM T59102 C0XM7N 59376046 IC50 = 118.4 nM T59102 C70WCP 59376053 IC50 = 15.6 nM T59102 C5IHG9 59376058 IC50 = 18 nM T59102 CTK90V 59376059 IC50 = 260.3 nM T59102 C7ZY5I 59376061 IC50 = 101.4 nM T59102 CFT69X 59376062 IC50 = 70.3 nM T59102 C7D0BF 59376072 IC50 = 13.2 nM T59102 CD0RP7 59376074 IC50 = 62.1 nM T59102 C3HXC7 59376075 IC50 = 19.3 nM T59102 CAY6H8 59376079 IC50 = 13.3 nM T59102 CCX2W0 59376082 IC50 = 160.6 nM T59102 CLH49Z 59790029 IC50 = 1 nM T59102 C9QRX3 60098131 IC50 = 310 nM T59102 CSZA16 60155724 IC50 > 3600 nM T59102 CU79HD 60202383 IC50 = 243 nM T59102 C9ZCT2 62705065 IC50 > 1000 nM T59102 CK6WO0 66552478 IC50 < 10000 nM T59102 C37NKO 67129970 IC50 > 10000 nM T59102 CK80LJ 67130050 IC50 > 10000 nM T59102 CA63QI 67219716 IC50 > 5000 nM T59102 CV63UL 67240318 IC50 > 10000 nM T59102 C7GRV2 68755406 IC50 > 10000 nM T59102 CCS20X 69063773 IC50 = 3 nM T59102 CEB12M 70681395 IC50 = 3 nM T59102 CH27DE 70681409 IC50 = 2 nM T59102 CN29RI 70681410 IC50 = 5 nM T59102 CG93IE 70683519 IC50 = 0.3 nM T59102 CXSN14 70685622 IC50 = 6 nM T59102 CL24MP 70687766 IC50 = 0.2 nM T59102 C51DHN 70689791 IC50 = 3 nM T59102 C6ITV3 70689792 IC50 = 0.9 nM T59102 CMLY63 70689816 IC50 = 0.5 nM T59102 C08ASR 70689830 IC50 = 4 nM T59102 C4TF3G 70691955 IC50 = 5 nM T59102 CTWD94 70691956 IC50 = 50 nM T59102 CIK5N2 70691957 IC50 = 10 nM T59102 C8RZP3 70691958 IC50 = 5 nM T59102 C0XRC9 70691981 IC50 = 3 nM T59102 C9RT8C 70693982 IC50 = 0.7 nM T59102 C2X1KJ 70694006 IC50 = 0.4 nM T59102 C54VLD 70694007 IC50 = 0.2 nM T59102 C6O3SM 70696108 IC50 = 50 nM T59102 CEBO91 71452977 IC50 > 10000 nM T59102 C9DIK2 71512060 IC50 = 2102 nM T59102 C6HF8S 71521082 IC50 = 35400 nM T59102 C9Z3AI 71521083 IC50 > 5000 nM T59102 C5OBF0 71525245 IC50 > 500000 nM T59102 CJX73B 71525246 IC50 > 500000 nM T59102 CCN90I 71525247 IC50 = 331500 nM T59102 CY6JA9 71525248 IC50 > 500000 nM T59102 CGQJ60 71525249 IC50 > 500000 nM T59102 CMKD15 71525283 IC50 = 89700 nM T59102 C3OJ6R 71525284 IC50 > 500000 nM T59102 CP5Q2U 71525285 IC50 = 430100 nM T59102 CZ8N0J 71525286 IC50 > 500000 nM T59102 CG31MI 71525287 IC50 > 500000 nM T59102 CRX81Q 71575642 IC50 = 408 nM T59102 CGK76E 71583411 IC50 > 200000 nM T59102 CB5WX0 71583412 IC50 > 200000 nM T59102 CI8K3T 71583527 IC50 = 196200 nM T59102 C6FGI0 71583528 IC50 > 200000 nM T59102 C3QGE7 71583529 IC50 = 172200 nM T59102 CS9HX7 71583530 IC50 = 70600 nM T59102 CQTZ32 71583531 IC50 > 200000 nM T59102 C0G5RS 71583532 IC50 > 200000 nM T59102 CVEY46 71583533 IC50 = 170800 nM T59102 CX6TR7 71583634 IC50 > 200000 nM T59102 CR15QP 71583635 IC50 = 196200 nM T59102 CZ31PU 71583657 IC50 > 10000 nM T59102 CU1IL6 71741204 IC50 > 100000 nM T59102 CN1GA3 71741327 IC50 > 100000 nM T59102 COS5D7 71741328 IC50 > 100000 nM T59102 C8PWZ0 71741329 IC50 > 100000 nM T59102 CT4XR9 71741332 IC50 > 50000 nM T59102 C4Q6FE 71815105 IC50 = 86.9 nM T59102 CJ9OX6 71815106 IC50 = 176.7 nM T59102 CCKL45 72191698 IC50 = 395.7 nM T59102 C60TUV 72737208 IC50 > 10000 nM T59102 CJ3WA6 72737404 IC50 > 10000 nM T59102 C8SIL6 73349435 IC50 = 1.42 nM T59102 CVNW01 73386831 IC50 > 1000 nM T59102 C2PAK9 73438493 IC50 = 1055 nM T59102 CBAT06 76071144 IC50 = 1083 nM T59102 CH8W7D 77461036 IC50 > 1000 nM T59102 CA65HB 78319164 IC50 = 20 nM T59102 CCJ43A 86302281 IC50 > 10000 nM T59102 CB5NJ4 86302541 IC50 = 4.6 nM T59102 CPG3A5 86302574 IC50 > 30000 nM T59102 C08WGI 86566799 IC50 = 16.3 nM T59102 C5S3YB 90645165 IC50 = 92.3 nM T59102 C6Q4DH 90645475 IC50 = 29.9 nM T59102 C89HTB 90645476 IC50 = 56.5 nM T59102 C9ASG1 90645478 IC50 = 27.1 nM T59102 COY53U 90645479 IC50 = 16.2 nM T59102 C48OSQ 90645480 IC50 = 23.1 nM T59102 CL8GW5 90645481 IC50 = 66.1 nM T59102 CL7SC6 90645482 IC50 = 28.3 nM T59102 CI3OD6 90645484 IC50 = 63.5 nM T59102 CX29IY 90655145 IC50 > 10000 nM T59102 C96DTL 90682879 IC50 = 21.9 nM T59102 CI97DL 102431709 IC50 = 19000 nM T59102 C09MIG 102431710 IC50 = 1500 nM T59102 C5HRO7 102431711 IC50 = 1400 nM T59102 CTGP06 117996541 IC50 > 10000 nM T59102 CY7BI2 118706214 IC50 > 10000 nM T59102 C2IN3C 118710236 IC50 = 8.1 nM T59102 CF2YR1 118710237 IC50 = 1.54 nM T59102 C4AHL2 118711367 IC50 = 5800 nM T59102 C46QUT 118717614 IC50 > 200000 nM T59102 CJC34Y 118717615 IC50 > 200000 nM T59102 CFEP93 118717616 IC50 > 200000 nM T59102 CEC4H0 118717617 IC50 > 200000 nM T59102 CU2TG3 118717618 IC50 > 200000 nM T59102 C5OL0W 118717619 IC50 > 200000 nM T59102 C3KLI5 118723185 IC50 = 500 nM T59102 C5UZ9X 118723186 IC50 = 4000 nM T59102 C3XV6L 118723187 IC50 > 100000 nM T59102 CLD41J 118723188 IC50 > 100000 nM T59102 C0H9YD 118723189 IC50 = 5000 nM T59102 CP8FW0 118723190 IC50 = 13000 nM T59102 CCV0H1 118723191 IC50 = 13000 nM T59102 C1J7QE 118723192 IC50 = 12000 nM T59102 CMHV05 118723193 IC50 = 32000 nM T59102 CRQY80 118723194 IC50 = 300 nM T59102 CVZM84 118723195 IC50 = 1000 nM T59102 CP8Z6I 118723196 IC50 = 14000 nM T59102 CI6HB3 118723197 IC50 = 56000 nM T59102 CVGE25 118723198 IC50 = 2000 nM T59102 C78BAF 118723199 IC50 = 9000 nM T59102 C02HAD 118723200 IC50 = 3000 nM T59102 CDAN63 118723201 IC50 = 26000 nM T59102 CL6T5K 118723202 IC50 = 1000 nM T59102 CDQ92V 118723203 IC50 = 8000 nM T59102 CV0B6M 118723204 IC50 = 2000 nM T59102 CX4E1N 118723205 IC50 = 1000 nM T59102 C8BU5O 118723206 IC50 = 2000 nM T59102 C2G1TN 118723207 IC50 = 7000 nM T59102 C1JO0D 118723208 IC50 = 22000 nM T59102 CYXF26 118723209 IC50 = 31000 nM T59102 C7JYP8 118723210 IC50 = 800 nM T59102 CV6HJ8 118723211 IC50 = 5000 nM T59102 CI6QA2 118723212 IC50 = 100 nM T59102 C3XKJ9 118723213 IC50 = 2000 nM T59102 CU1B5W 118723214 IC50 = 19000 nM T59102 CD5HK1 118723215 IC50 = 8000 nM T59102 CU06YS 118723216 IC50 > 100000 nM T59102 CWYF91 118729842 IC50 = 40.4 nM T59102 CR54XL 118729843 IC50 = 66.1 nM T59102 CF3X9J 118729844 IC50 = 166.3 nM T59102 CT3Q6C 118729845 IC50 = 50.1 nM T59102 C1QWK6 118729846 IC50 = 24.6 nM T59102 CWUA61 118729847 IC50 = 25 nM T59102 C63CDP 118729848 IC50 = 73.2 nM T59102 C1WB7L 118729849 IC50 = 198 nM T59102 C8A7ZT 118729850 IC50 = 58.2 nM T59102 C9WDF4 118729851 IC50 = 84 nM T59102 CT08EZ 118729852 IC50 = 132 nM T59102 C08KEM 122179540 IC50 = 2000 nM T59102 CG0RP7 122179547 IC50 = 2200 nM T59102 C1A0SQ 122179548 IC50 = 4600 nM T59102 C4X7SD 122192466 IC50 = 1982 nM T59102 CNX0Q2 122193763 IC50 = 850 nM T59102 CWV0C3 122193764 IC50 = 2120 nM T59102 CSG98Y 122193765 IC50 = 2820 nM T59102 CCLQ75 122193769 IC50 = 320 nM T59102 CXDR48 122193770 IC50 = 570 nM T59102 CPA8C5 122193773 IC50 = 2300 nM T59102 CY30FL 123752658 IC50 = 5.5 nM T59102 C8KXV1 127025843 IC50 > 1000 nM T59102 C1XD6R 127029809 IC50 = 526.5 nM T59102 CI1E5W 127029864 IC50 = 4.57 nM T59102 CKS28E 127034802 IC50 = 64.2 nM T59102 CKX40V 127037812 IC50 = 223.9 nM T59102 C70RUP 127038480 IC50 > 10000 nM T59102 C3WCN8 127041777 IC50 > 10000 nM T59102 CC58IQ 127043948 IC50 = 120 nM T59102 CHK16Q 127045929 IC50 > 1000 nM T59102 CY3J0C 127047591 IC50 > 1000 nM T59102 CF5D2Y 129318936 IC50 = 6115 nM T59102 C0FM1R 130196825 IC50 = 392 nM T59102 CUO0C5 132156633 IC50 > 10000 nM T59102 C6OMB1 132204257 IC50 = 606 nM T59102 C6ROQ3 132546210 IC50 = 80 nM T59102 CJ04HZ 132585195 IC50 < 1 nM T59102 CERS64 132937256 IC50 = 26197 nM T59102 CN9SD7 132942957 IC50 = 51.4 nM T59102 CMP2S9 132942958 IC50 = 62.2 nM T59102 CN35SO 134146628 IC50 > 1000 nM T59102 CIK38Q 134229735 IC50 = 63.4 nM T59102 CYL5V1 134694986 IC50 > 30000 nM T59102 CLCO61 135398510 EC50 = 51 nM T59102 CN5T7W 135400982 IC50 = 12 nM T59102 CVJ07T 135402853 IC50 = 70 nM T59102 CBK6I2 135407156 IC50 = 30 nM T59102 CMVS34 135410282 IC50 = 10 nM T59102 CUT52Q 135421574 IC50 = 19000 nM T59102 CK9D4A 135428921 IC50 = 4500 nM T59102 C8X5SV 135433815 IC50 = 20 nM T59102 CNZ04G 135453357 IC50 = 4 nM T59102 CS63IO 135476717 IC50 = 65 nM T59102 C2MAC7 135536640 IC50 > 100000 nM T59102 CW08GF 135674125 IC50 = 70 nM T59102 CLS64T 135674129 IC50 = 0.9 nM T59102 C54ABM 135674133 IC50 = 0.3 nM T59102 CM7YH4 135674136 IC50 = 5 nM T59102 C1WSO7 135674140 IC50 = 130 nM T59102 CA0Y7V 135674142 IC50 = 5 nM T59102 CM90FP 135674144 IC50 = 0.9 nM T59102 C3CP1X 135674147 IC50 = 0.3 nM T59102 CBSV42 135674149 IC50 = 5 nM T59102 C1NTB0 135674153 IC50 = 2 nM T59102 CID0W9 135674167 IC50 = 0.1 nM T59102 C1DL9J 135674173 IC50 = 30 nM T59102 CO89UX 135674193 IC50 = 8 nM T59102 C2H3XB 135926086 IC50 = 2 nM T59102 C7BES6 135926087 IC50 = 2 nM T59102 CNTK81 135926088 IC50 = 7 nM T59102 CQ64OH 135926089 IC50 = 39 nM T59102 CXG7O4 135926090 IC50 = 0.1 nM T59102 CN4FG3 135926091 IC50 = 14 nM T59102 C7NZU3 135926094 IC50 > 25000 nM T59102 CL6HQ4 135926104 IC50 = 1 nM T59102 CE37KQ 135926113 IC50 = 0.7 nM T59102 C1ZRT7 135926114 IC50 = 1 nM T59102 CU5W2V 135926115 IC50 = 7 nM T59102 C1D3EW 135926116 IC50 = 0.6 nM T59102 C2PAV1 135971426 IC50 = 10000 nM T59102 CHA4N2 136013680 IC50 > 10 nM T59102 CLN6Y8 136026516 IC50 > 100000 nM T59102 CG1R7B 136087060 IC50 = 7000 nM T59102 C5QZ4H 136126664 IC50 = 1100 nM T59102 CB8RX0 136126665 IC50 = 0.2 nM T59102 CZ7EX0 136183413 IC50 = 3200 nM T59102 CDT7E4 136211077 IC50 > 1000 nM T59102 C9RE8D 136215817 IC50 = 530.6 nM T59102 C1YUD0 136219394 IC50 > 10 nM T59102 CIU8W3 136254389 IC50 > 10 nM T59102 C35MBU 136299423 IC50 = 45 nM T59102 C0W8KA 136299435 IC50 = 4.3 nM T59102 C5G4ES 136299436 IC50 = 3.2 nM T59102 C83OXU 137007054 IC50 = 12000 nM T59102 CCM42D 137249694 IC50 = 14.3 nM T59102 C25ERN 137631967 IC50 = 1 nM T59102 CFUY16 137633842 IC50 > 200000 nM T59102 CNX0F9 137634126 IC50 = 106.2 nM T59102 CHC70D 137634143 IC50 = 3.26 nM T59102 CI1E8V 137634241 IC50 = 5190 nM T59102 C85WBP 137634338 IC50 = 9 nM T59102 CAD3C5 137634686 IC50 = 45.52 nM T59102 CS23KQ 137635618 IC50 = 90100 nM T59102 C5JD9N 137635898 IC50 = 10.3 nM T59102 CK5Y3P 137635915 IC50 = 65.24 nM T59102 C06JRX 137637094 IC50 > 10 nM T59102 CU24QC 137638448 IC50 = 90.3 nM T59102 CO9D4W 137639407 IC50 = 31.36 nM T59102 C3UBE2 137639638 IC50 > 200 nM T59102 CU8YX6 137643005 IC50 = 58200 nM T59102 C2T6FV 137644825 IC50 = 29.79 nM T59102 C1DK0P 137651391 IC50 = 1 nM T59102 C5F3LP 137651946 IC50 = 83.17 nM T59102 CQUY83 137652218 IC50 > 200000 nM T59102 C9JT1N 137655519 IC50 = 60500 nM T59102 C9TEU1 137655771 IC50 = 27.11 nM T59102 CKVO51 137657233 IC50 = 30.2 nM T59102 CV5H3Z 137657932 IC50 > 100 nM T59102 CQMB10 137658515 IC50 = 197 nM T59102 C7IVT9 137658762 IC50 > 200 nM T59102 CQE9M4 137661156 IC50 = 67.85 nM T59102 CM0N3T 137661420 IC50 = 7.2 nM T59102 CT43IF 137661858 IC50 = 8.1 nM T59102 CIWG23 138393067 IC50 = 88 nM T59102 C07EKN 138454794 IC50 = 2075 nM T59102 C5LQU9 138479230 IC50 = 673.6 nM T59102 CSRI06 138547901 IC50 > 1000 nM T59102 CUXO19 138617501 IC50 > 1000 nM T59102 C6AK0N 139030518 IC50 = 97 nM T59102 C34CKN 141523354 IC50 = 19.46 nM T59102 CB3Z1W 145949428 IC50 = 180 nM T59102 CCM27G 145949662 IC50 = 64.6 nM T59102 CVJS01 145949677 IC50 = 12 nM T59102 CWQA26 145949916 IC50 = 34.3 nM T59102 CYF32C 145950953 IC50 = 15 nM T59102 CRXJ25 145951211 IC50 = 91 nM T59102 C4LBC0 145951650 IC50 = 116.2 nM T59102 CR9LH4 145952520 IC50 = 92.7 nM T59102 CC72WG 145953067 IC50 = 7800 nM T59102 C60XZR 145953297 IC50 = 19 nM T59102 CSLC73 145953358 IC50 = 44.2 nM T59102 CAL30B 145953560 IC50 = 15 nM T59102 C0V8SM 145954139 IC50 = 25 nM T59102 CDRQ06 145955547 IC50 = 45.5 nM T59102 C8VN1Y 145955561 IC50 = 27 nM T59102 C2O9XD 145955651 IC50 = 91.7 nM T59102 C1IX5N 145956333 IC50 = 22 nM T59102 C6ZNJ1 145956488 IC50 = 34 nM T59102 CLZH04 145956490 IC50 = 39 nM T59102 C5VSC7 145956704 IC50 = 177 nM T59102 CY69RH 145956768 IC50 = 49.2 nM T59102 CIW0V9 145956964 IC50 = 241.6 nM T59102 CB74GR 145957221 IC50 = 24 nM T59102 CB1MI9 145957910 IC50 = 4.5 nM T59102 CS47UF 145958497 IC50 = 14 nM T59102 CRVO52 145960991 IC50 > 500 nM T59102 CV4M1Z 145961849 IC50 = 60.7 nM T59102 C9PKU6 145963750 IC50 = 5.3 nM T59102 CTUF34 145966712 IC50 = 111 nM T59102 C4OD9Q 145967187 IC50 = 214.5 nM T59102 CNVT54 145971746 IC50 = 61 nM T59102 C3Q4XM 145972183 IC50 = 13 nM T59102 C71ZJX 145972445 IC50 = 135.1 nM T59102 CG8R0P 145972697 IC50 = 1.5 nM T59102 C74TYP 145975351 IC50 = 482.1 nM T59102 CCS92I 145982511 IC50 = 510 nM T59102 CWE21T 145982588 IC50 = 3250 nM T59102 CC12YA 145982666 IC50 = 57.8 nM T59102 CF4BO8 145982785 IC50 = 28.9 nM T59102 CM6ZS7 145982824 IC50 = 63 nM T59102 CZ3CG9 145982825 IC50 = 1260 nM T59102 CF28AU 145983389 IC50 = 42.6 nM T59102 CRL19G 145983447 IC50 = 40 nM T59102 C48UZH 145983504 IC50 = 2230 nM T59102 C8BZC5 145983753 IC50 = 20 nM T59102 CD5L8O 145983778 IC50 > 200 nM T59102 CNK7I9 145984104 IC50 = 3520 nM T59102 C4C2OM 145984258 IC50 = 8 nM T59102 C9DHL3 145984282 IC50 = 3780 nM T59102 CVT02P 145984555 IC50 = 20 nM T59102 CHW8E5 145984671 IC50 = 1230 nM T59102 CYG42V 145984818 IC50 > 200 nM T59102 CFS7D5 145984941 IC50 > 200 nM T59102 C05IMJ 145984942 IC50 = 38.9 nM T59102 C9Q5VI 145985608 IC50 = 820 nM T59102 CA2TW8 145985737 IC50 = 290 nM T59102 CS9C8J 145986155 IC50 > 200 nM T59102 C1Y5MO 145987062 IC50 = 1.81 nM T59102 CI85EU 145998085 IC50 = 1013 nM T59102 C2MD1Q 155513187 IC50 > 10000 nM T59102 C86HPW 155518524 IC50 = 81000 nM T59102 CU6Z5O 155520650 IC50 = 150 nM T59102 CY6NE1 155523855 IC50 = 100 nM T59102 CRP7Q6 155525519 IC50 = 110 nM T59102 CTD5R7 155528337 IC50 = 450 nM T59102 CLEJ03 155529517 IC50 = 230 nM T59102 CS69CA 155532132 IC50 = 25.3 nM T59102 C3NZO0 155533789 IC50 = 90 nM T59102 C2DJ0A 155534253 IC50 = 2010 nM T59102 C37RFQ 155534994 IC50 = 1590 nM T59102 CE46SL 155540854 IC50 > 30000 nM T59102 C5O4JM 155540856 IC50 > 30000 nM T59102 C7SF2C 155547229 IC50 = 356 nM T59102 C6URZ7 155550475 IC50 = 1820 nM T59102 CGVU70 155554426 IC50 > 30000 nM T59102 CUA73V 155555832 IC50 = 330 nM T59102 C8L6PM 155561965 IC50 = 3790 nM T59102 C81JZW 155563388 IC50 = 390 nM T59102 CM23DI 155565660 IC50 = 1290 nM T59102 CK10HA 155568167 IC50 = 3640 nM T59102 CBWO68 49800164 IC50 = 28 nM T59102 D00ATA 5908088 IC50 = 12000 nM T59102 D00GVV 5329155 IC50 = 920 nM T59102 D02BXJ 46864270 IC50 = 2.6 nM T59102 D04FNY 25195216 IC50 = 40 nM T59102 D05NKG 16760286 IC50 = 316.23 nM T59102 D05WTI 11550535 IC50 = 317 nM T59102 D06QWO 14824655 IC50 > 10 ug.mL-1 T59102 D07IHM 9823787 IC50 > 10000 nM T59102 D07OSK 6419834 IC50 = 4000 nM T59102 D09HVH 135566652 IC50 > 10 nM T59102 D09LPL 5329103 IC50 = 3 nM T59102 D09QBA 23378546 IC50 > 10000 nM T59102 D09TNR 9850161 IC50 = 69 nM T59102 D0A1CM 5281855 IC50 = 1300 nM T59102 D0A4XJ 5289418 IC50 = 510 nM T59102 D0BW4G 10907042 IC50 = 130 nM T59102 D0C2GE 67161540 IC50 = 1.3 nM T59102 D0D6MH 11617559 IC50 > 10000 nM T59102 D0EE6A 6398883 IC50 = 640 nM T59102 D0G3SZ 6918469 IC50 = 5.9 ug.mL-1 T59102 D0H1OK 11562302 Ki = 2090 nM T59102 D0HE0E 5941540 IC50 = 5100 nM T59102 D0I3XZ 11601743 IC50 = 171 nM T59102 D0L3FK 5289419 IC50 > 10000 nM T59102 D0M4QA 56935577 IC50 = 10.1 nM T59102 D0R2WK 16038120 IC50 = 3220 nM T59102 D0U3WQ 9817165 IC50 = 90 nM T59102 D0UN9O 3385203 IC50 = 1000 nM T59102 D0X1RH 16051023 IC50 = 420 nM T59102 D0XS9E 5330535 IC50 = 90 nM T59102 D0YE1X 9927943 IC50 = 30 nM T59102 D0YZ7H 9797370 IC50 = 3 nM T59102 D0Z7TM 22273644 IC50 > 2000 nM T85272 D03DAP 3356 IC50 = 209000 nM T85272 D04OSE 4485 IC50 = 96000 nM T85272 D08YIN 1727 IC50 = 89000 nM T85272 D0OB1J 39186 IC50 = 144000 nM T85272 D0U5CE 1548943 IC50 = 29000 nM T85272 D0K9IF 71666749 IC50 > 30000 nM T85272 C29SPL 5867 EC50 = 33000 nM T85272 C6HA8E 5388709 IC50 > 30000 nM T85272 C8W2QA 6439099 IC50 > 30000 nM T85272 C8NM2I 11538313 EC50 = 7000 nM T85272 CA5W9R 11618060 EC50 = 1200 nM T85272 CLT3Z7 11695929 EC50 = 1700 nM T85272 CW9V0Y 13088125 EC50 = 6000 nM T85272 C8JA3E 13703975 EC50 = 4300 nM T85272 C91QFN 25019282 IC50 = 2660 nM T85272 CQSZ72 90675942 IC50 > 30000 nM T85272 CTBD74 90675943 IC50 > 30000 nM T85272 CM12LR 102597975 IC50 > 30000 nM T85272 CQJ49Y 122187245 IC50 = 0.0067 nM T85272 CSW57U 122187246 IC50 = 0.0077 nM T85272 C98BUE 122187247 IC50 = 0.0034 nM T85272 CVT7A6 122187248 IC50 = 0.0027 nM T85272 CI9ZH1 122187249 IC50 = 0.0078 nM T85272 CHJ75V 122187250 IC50 = 0.0095 nM T85272 C20TPX 122187251 IC50 = 0.0028 nM T85272 CQ17ZP 122187252 IC50 = 0.011 nM T85272 C2XUA5 122187253 IC50 = 0.308 nM T85272 CQTJ57 122187272 IC50 = 0.0078 nM T85272 CX2YG6 122187273 IC50 = 0.0181 nM T85272 C4CLN5 122187274 IC50 > 3.333 nM T85272 CF5M8V 122187275 IC50 = 0.49 nM T85272 C24MEW 122187276 IC50 > 3.333 nM T85272 CI7VL5 122187277 IC50 > 3.333 nM T85272 COX2P3 122187278 IC50 = 0.014 nM T85272 CY9RL0 122187279 IC50 = 0.02 nM T85272 CT5B4D 122187280 IC50 = 0.028 nM T85272 C42SZA 122187281 IC50 = 1.8 nM T85272 C6S3XG 122187282 IC50 = 0.0018 nM T85272 C0YG3Z 122187283 IC50 = 0.0057 nM T85272 C1F5PE 122187284 IC50 = 0.0023 nM T85272 C26VHJ 122187285 IC50 = 0.0049 nM T85272 C24JCI 122187286 IC50 = 0.0083 nM T85272 CW4SU9 122187287 IC50 = 0.001 nM T85272 CT0GS6 122187288 IC50 = 0.007 nM T85272 CCO3Y2 122187289 IC50 = 3.279 nM T85272 C1ENW4 122187290 IC50 = 0.046 nM T85272 CFH36G 122187291 IC50 = 0.0172 nM T85272 C3CY5N 122187292 IC50 = 0.004 nM T85272 CY69QI 122187293 IC50 = 0.0027 nM T85272 C05WQZ 122187294 IC50 = 0.003 nM T85272 C1LW9V 122187295 IC50 = 0.0195 nM T85272 CBMT85 122187296 IC50 = 0.0018 nM T85272 C8AKN9 122187297 IC50 = 0.0154 nM T85272 CDM71F 122187298 IC50 = 0.055 nM T85272 CCM08N 122187299 IC50 = 0.0038 nM T85272 C7V2TW 122187300 IC50 = 0.0028 nM T85272 C81QSJ 122187301 IC50 > 3.333 nM T85272 C1IPG9 122187302 IC50 = 0.0324 nM T85272 C0RE2W 122187303 IC50 > 3.333 nM T85272 C9JDM3 122187304 IC50 > 3.333 nM T85272 C5QXR6 122187305 IC50 = 0.0087 nM T85272 C50RMQ 122187306 IC50 = 0.0018 nM T85272 C5Z9PU 122187307 IC50 = 0.07 nM T85272 CT0V4W 122187308 IC50 > 3.333 nM T85272 CX06CZ 122187309 IC50 = 0.008 nM T85272 CK9T7F 122187310 IC50 = 0.59 nM T85272 CC2LE0 122187311 IC50 = 0.0036 nM T85272 CS34VD 122187312 IC50 = 0.002 nM T85272 CIU9T5 122187313 IC50 = 0.0031 nM T85272 CS8QW7 122187314 IC50 = 0.0042 nM T85272 CID97N 122187315 IC50 = 0.458 nM T85272 CZ08GP 122187316 IC50 = 0.0026 nM T85272 C0P6IC 122187317 IC50 > 3.333 nM T85272 CY7M0F 122187318 IC50 = 0.005 nM T85272 CQZK10 122187319 IC50 = 0.0033 nM T85272 C62FDT 122187320 IC50 = 0.0024 nM T85272 C3QZY1 122187321 IC50 = 0.0044 nM T85272 C8B4YL 122187322 IC50 = 0.005 nM T85272 CWV12K 122187323 IC50 = 0.0527 nM T85272 CWVP15 122187324 IC50 = 2.342 nM T85272 CEW35A 122187325 IC50 = 0.0017 nM T85272 CP43GQ 122187326 IC50 = 0.0021 nM T85272 CH46BC 122187327 IC50 = 0.04 nM T85272 C6KW2B 122187328 IC50 = 0.004 nM T85272 C87MGD 122187329 IC50 = 0.0028 nM T85272 C0U9QN 122187330 IC50 = 0.0335 nM T85272 CH4G1L 122187331 IC50 = 0.075 nM T85272 C4ZR9M 122187332 IC50 = 0.266 nM T85272 CM8A1Y 122187333 IC50 = 0.174 nM T85272 CU3IE9 122187334 IC50 = 0.005 nM T85272 CYN12K 122187335 IC50 = 0.0051 nM T85272 CDE52G 122187336 IC50 = 0.74 nM T85272 CZH25J 122187337 IC50 = 0.011 nM T85272 CQP1R4 122187338 IC50 = 0.6 nM T85272 C3QS0A 122187339 IC50 = 9.5 nM T85272 CAFO71 122187340 IC50 = 0.015 nM T85272 CNYJ15 122187341 IC50 = 29.26 nM T85272 CY62QW 122187342 IC50 = 13.22 nM T85272 CCV2G0 122187343 IC50 > 33.33 nM T85272 C0Z8JH 122187344 IC50 = 0.014 nM T85272 CVT8Z7 122187345 IC50 = 0.847 nM T85272 C2YI7W 122187346 IC50 = 0.214 nM T85272 CO7MU2 122187445 IC50 = 0.002 nM T85272 C8QN9Z 122187446 IC50 = 0.0068 nM T85272 C09YUX 122187447 IC50 = 0.005 nM T85272 C8I6TF 122187448 IC50 = 0.0022 nM T85272 CR68ZK 122187449 IC50 = 0.0035 nM T85272 CTY96B 122187450 IC50 = 0.0053 nM T85272 C4WG0M 122187451 IC50 = 0.0182 nM T85272 CLS4H7 122187452 IC50 = 0.0014 nM T85272 CM23CQ 122187453 IC50 = 0.76 nM T85272 CJF8X1 122187454 IC50 > 3.333 nM T85272 C54PSK 122187455 IC50 = 0.005 nM T85272 CGS5Q1 122187456 IC50 = 0.0014 nM T85272 CW0MH4 122187457 IC50 = 0.0011 nM T85272 CXAV52 122187458 IC50 = 0.0034 nM T85272 C3D8EQ 122187459 IC50 = 0.446 nM T85272 CBUT59 122187460 IC50 = 0.005 nM T85272 C1XL3M 122187461 IC50 = 0.004 nM T85272 CBS95M 122187462 IC50 = 0.005 nM T85272 CY79JC 122187463 IC50 = 0.0037 nM T85272 CAY0P4 122187464 IC50 = 0.006 nM T85272 CRQ98D 122187465 IC50 = 0.006 nM T85272 CXP98T 122187466 IC50 = 0.0042 nM T85272 C5TJU8 122187467 IC50 > 3.333 nM T85272 CP7C2I 122187468 IC50 = 0.028 nM T85272 CKC0L8 122187469 IC50 = 0.305 nM T85272 CV3T2C 122187470 IC50 = 0.011 nM T85272 CN5OQ2 122187471 IC50 = 0.0009 nM T85272 CI0J4A 122187472 IC50 = 0.0274 nM T85272 CM14KC 122187473 IC50 = 0.0157 nM T85272 COFI26 122187474 IC50 = 0.0489 nM T85272 CTXG58 122187475 IC50 = 0.0102 nM T85272 CZWG59 122187476 IC50 > 3.333 nM T85272 C1TVY5 122187477 IC50 = 0.0033 nM T85272 CS6FK8 122187478 IC50 > 3.333 nM T85272 CJC21F 122187479 IC50 = 0.0262 nM T85272 C3ZE4Y 122187480 IC50 > 3.333 nM T85272 CS0U8H 122187481 IC50 > 3.333 nM T85272 CY0NV5 122187482 IC50 = 0.0091 nM T85272 C8SHE5 122187483 IC50 = 1.018 nM T85272 CHYI14 122187484 IC50 = 2.42 nM T85272 CEH14V 122187485 IC50 > 3.333 nM T85272 CG98KU 122187486 IC50 = 0.0032 nM T85272 C3P8WN 122187487 IC50 = 0.0061 nM T85272 C9MJ2K 122187488 IC50 = 0.0061 nM T85272 C7J0YH 122187489 IC50 = 0.0044 nM T85272 C4NYT7 122187490 IC50 = 0.04 nM T85272 CMT25I 122187491 IC50 = 0.0015 nM T85272 CQEV80 122187492 IC50 = 0.0076 nM T85272 CY07HP 122187493 IC50 = 1.2 nM T85272 CD0EU3 122187494 IC50 = 0.0256 nM T85272 CQZ0R1 122187495 IC50 = 0.032 nM T85272 CZU4N2 122187496 IC50 = 0.0073 nM T85272 CITK91 122187497 IC50 = 0.0059 nM T85272 C69JKA 122187498 IC50 = 0.0042 nM T85272 C6R5CY 122187499 IC50 = 0.029 nM T85272 CM87YE 122187500 IC50 = 0.0045 nM T85272 CP4GJ7 122187501 IC50 = 0.051 nM T85272 CB14ES 122187502 IC50 = 0.004 nM T85272 CEGB98 122187503 IC50 = 0.042 nM T85272 CU61JG 137651545 IC50 = 13000 nM T85272 CW9P6A 145964460 IC50 > 30000 nM T85272 CQR49Z 145965116 IC50 > 30000 nM T85272 CR6L2G 145967358 IC50 > 30000 nM T85272 CHXE25 145978207 IC50 > 30000 nM T85272 D06PZZ 5413 IC50 = 30000 nM T85272 D08BMM 6312649 IC50 > 30000 nM T85272 D0R9CF 11302540 IC50 = 250 nM T96736 CR57DL 50803848 IC50 = 35000 nM T96736 CP79TH 52931882 IC50 = 2580 nM T96736 CPE79U 52931883 IC50 = 3280 nM T96736 C9LGO3 52931939 IC50 = 2620 nM T96736 C92SRX 52931998 IC50 = 1510 nM T96736 C5F1IT 52932001 IC50 = 2050 nM T96736 CWFG81 52932003 IC50 = 1680 nM T96736 C65DNB 52932059 IC50 = 1240 nM T96736 C06LVX 53363853 IC50 = 2090 nM T96736 C3QGZ1 53364100 IC50 = 3000 nM T96736 CXYI14 71681394 IC50 = 9200 nM T96736 COBN97 71681395 IC50 = 10000 nM T96736 CR5BQ2 71681396 IC50 = 31000 nM T96736 C6E8TM 71681562 IC50 = 9900 nM T96736 C7ITA6 71681563 IC50 = 27000 nM T96736 C9KP1U 71681564 IC50 = 26000 nM T96736 CE6P5O 71681565 IC50 = 33000 nM T96736 CH4F1V 71681566 IC50 = 33000 nM T96736 CA2GQ5 71681720 IC50 = 35000 nM T96736 CP8UN5 71681721 IC50 = 43000 nM T96736 C6O8VG 71681722 IC50 = 51000 nM T96736 C3WU8P 71681723 IC50 = 67000 nM T96736 CA68PI 71681724 IC50 = 78000 nM T96736 C0TKW7 71682046 IC50 = 1500 nM T96736 CGJ18W 71682047 IC50 = 1600 nM T96736 CGMO97 71682048 IC50 = 2300 nM T96736 C4QA6W 71682049 IC50 = 5600 nM T96736 CY63JH 71682050 IC50 = 6100 nM T96736 C2QH9Y 71682204 IC50 = 8100 nM T96736 CS45BO 71682205 IC50 = 11000 nM T96736 CE87JT 71682206 IC50 = 12000 nM T96736 C5KR2M 71682207 IC50 = 12000 nM T96736 CKG6I5 71682208 IC50 = 26000 nM T96736 C4MDP1 71682354 IC50 = 30000 nM T96736 C1H9AY 71682355 IC50 = 32000 nM T96736 CB9J7C 71682356 IC50 = 32000 nM T96736 C0X4DB 71682357 IC50 = 66000 nM T96736 CPQ8K0 71682358 IC50 = 76000 nM T96736 CM82DF 71682662 IC50 = 21000 nM T96736 C5XR3L 71682663 IC50 = 7400 nM T96736 C96MSZ 71682815 IC50 = 10000 nM T96736 C0IE1G 73349029 IC50 = 4700 nM T96736 D0I3KR 71681561 IC50 = 5300 nM T96736 D0Y9BU 46190808 IC50 = 9800 nM T86808 CL2Q6J 44178077 IC50 > 100000 nM T86808 C0BQC4 44586265 IC50 = 2200 nM T86808 C2IML9 58580486 IC50 = 460 nM T86808 D0K1NM 20541332 IC50 > 100000 nM T55398 D0OB0F 5328940 IC50 = 574 nM T55398 D03LWG 53235510 IC50 > 10000 nM T55398 D07EHV 44814409 IC50 > 10000 nM T55398 D07NUL 118414016 IC50 = 2 nM T55398 D0E3TC 44259 IC50 = 4.21 nM T55398 D0T3ME 156422 IC50 > 30000 nM T55398 CGEW10 1247796 IC50 = 2200 nM T55398 CJ3U9Y 2728161 IC50 = 55000 nM T55398 CF6WI5 2824236 IC50 = 2800 nM T55398 C1KY3I 4455946 IC50 = 12000 nM T55398 CRC65X 9863786 IC50 > 30000 nM T55398 C5UG6X 10114595 Ki = 0.48 nM T55398 C8K9HL 10142476 Ki = 0.42 nM T55398 C4RNU9 10184123 Ki = 0.5 nM T55398 CN37YZ 10207985 Ki = 0.34 nM T55398 C8BHJ3 10226185 Ki = 8.2 nM T55398 C78SMB 10227510 Ki = 2.8 nM T55398 CXN06I 10227557 Ki = 2.8 nM T55398 C0SR5Y 10278151 Ki = 0.7 nM T55398 CBOP58 11293798 Ki > 10000 nM T55398 C26BZX 11362471 Ki > 10000 nM T55398 CWXB93 11397177 Ki > 10000 nM T55398 CTG83F 11539329 Ki > 9900 nM T55398 CACS26 11561968 Ki > 4000 nM T55398 CMIL86 11590363 Ki > 9900 nM T55398 C9T6SC 11640926 Ki > 9900 nM T55398 CU0E8O 11690457 Ki = 1900 nM T55398 CB0AP2 11705863 Ki > 4000 nM T55398 CE2VU0 11987888 Ki = 1.2 nM T55398 CFPW41 16007116 Ki > 9900 nM T55398 CST43D 21899140 Ki = 6.5 nM T55398 CM4F0B 21899142 Ki = 1.3 nM T55398 CT46EH 21899147 IC50 = 8000 nM T55398 C7YG1N 24759534 IC50 = 210 nM T55398 CIN29Y 24801862 IC50 = 400 nM T55398 CZ12SD 24801863 IC50 = 3000 nM T55398 CZJ9P4 24857834 IC50 = 70 nM T55398 C3E5XY 24857850 IC50 = 420 nM T55398 CLZ23U 24951610 IC50 = 1100 nM T55398 C2KY1G 25094210 IC50 = 167 nM T55398 CGT1W6 25144294 IC50 = 56 nM T55398 CU7VR0 25144732 IC50 = 8 nM T55398 C6BWZ8 25145145 IC50 = 1000 nM T55398 CA75YC 25169380 IC50 = 6 nM T55398 CC3BU0 25169381 IC50 = 4 nM T55398 CFB65H 25169382 IC50 = 6 nM T55398 CRXS80 25169384 IC50 = 9 nM T55398 CC71QJ 27666048 IC50 > 100000 nM T55398 CTA08W 41420877 IC50 = 2000 nM T55398 CO6HU7 44178069 IC50 = 1142 nM T55398 C8KNA3 44219632 Ki > 4000 nM T55398 C0VIX4 44219633 Ki = 2300 nM T55398 CZH6G2 44412152 IC50 > 30000 nM T55398 C1OQP6 44412156 IC50 = 1500 nM T55398 CJR94S 44412164 IC50 > 30000 nM T55398 COZ5X9 44412166 IC50 = 25000 nM T55398 CU7Q3F 44412167 IC50 = 4000 nM T55398 CU0T2G 44412174 IC50 = 1000 nM T55398 C0V4FU 44412178 IC50 = 550 nM T55398 CIF5C1 44412201 IC50 = 1000 nM T55398 CCY3L4 44412220 IC50 = 20000 nM T55398 CR7Y9K 44412242 IC50 = 30000 nM T55398 C4UOZ2 44412243 IC50 = 6000 nM T55398 CGJ61S 44412251 Ki = 4500 nM T55398 C18ZMY 44412252 IC50 = 800 nM T55398 CM6X1B 44412253 IC50 = 2000 nM T55398 C6TN3O 44412266 IC50 = 1000 nM T55398 CD2W6N 44412267 IC50 = 2000 nM T55398 CRB74Z 44412281 IC50 = 400 nM T55398 C0R2LO 44412325 IC50 = 30000 nM T55398 CA0MI2 44412326 IC50 = 400 nM T55398 CH7M4G 44412327 IC50 = 1000 nM T55398 C35CLR 44412343 IC50 = 150 nM T55398 C7XE0D 44412352 IC50 = 4000 nM T55398 CUV9B8 44412391 IC50 = 6500 nM T55398 CH6F7D 44412392 IC50 = 2000 nM T55398 CG3LU0 44412407 IC50 = 30000 nM T55398 CZ16BF 44412434 IC50 = 4000 nM T55398 CA48QG 44412435 IC50 = 3000 nM T55398 C20AUC 44412442 IC50 = 500 nM T55398 C6N1MJ 44412480 IC50 = 3000 nM T55398 C6O0TZ 44412492 IC50 = 6500 nM T55398 CRK51G 44448764 IC50 = 39 nM T55398 CKI6S2 44448795 IC50 = 6900 nM T55398 C1HB0N 44448797 IC50 = 313 nM T55398 C7GA2S 44448798 IC50 = 3030 nM T55398 CTGL39 44448828 IC50 = 225 nM T55398 CSAH90 44448865 IC50 = 1300 nM T55398 CDWX21 44448867 IC50 = 914 nM T55398 CXV8T5 44448904 IC50 = 497 nM T55398 C3DP0G 44448905 IC50 = 8100 nM T55398 CAQ4T1 44448906 IC50 = 433 nM T55398 CO7Y6K 44448908 IC50 = 1134 nM T55398 COY50K 44448910 IC50 = 1085 nM T55398 CL28QE 44448912 IC50 = 10 nM T55398 CVQ74G 44448939 IC50 = 49 nM T55398 CIUF03 44448940 IC50 = 1156 nM T55398 C28SLH 44448941 IC50 = 5 nM T55398 C47GQS 44448942 IC50 = 263 nM T55398 CCV97Y 44448943 IC50 = 166 nM T55398 CHCN76 44448970 IC50 = 2 nM T55398 C3YM1B 44448971 IC50 = 63 nM T55398 C4S5TP 44448972 IC50 = 112 nM T55398 CV5F0Q 44448973 IC50 = 7 nM T55398 CX8PM6 44448975 IC50 = 3 nM T55398 CH61MQ 44449000 IC50 = 8 nM T55398 C3C2TM 44449002 IC50 = 181 nM T55398 CT3B1M 44449003 IC50 = 208 nM T55398 CE07NB 44449025 IC50 = 15 nM T55398 C5X0LI 44449050 IC50 = 1 nM T55398 CZ3V1X 44449078 IC50 = 35 nM T55398 C0SQE3 44449102 IC50 = 216 nM T55398 CK6E5J 44449122 IC50 = 95 nM T55398 CT7U9G 44449126 IC50 = 7 nM T55398 C37YOA 44449160 IC50 = 487 nM T55398 CXL76B 44449162 IC50 = 535 nM T55398 CSRC92 44449189 IC50 = 1880 nM T55398 CQ5I9D 44449190 IC50 = 126 nM T55398 C3DU4B 44449218 IC50 = 19 nM T55398 C64YUV 44449221 IC50 = 545 nM T55398 C1G4DC 44449335 IC50 = 710 nM T55398 C0CR1V 44449336 IC50 = 660 nM T55398 C1W9XR 44449364 IC50 = 1600 nM T55398 CMC7U0 44449365 IC50 > 10000 nM T55398 C2DCP7 44449366 IC50 > 10000 nM T55398 CP6R3S 44449367 IC50 > 10000 nM T55398 C6IHR2 44449391 IC50 = 3400 nM T55398 CJ68ZB 44449392 IC50 = 160 nM T55398 CZJ8U5 44449393 IC50 = 350 nM T55398 CZYR60 44449394 IC50 = 1200 nM T55398 C2SO6L 44449424 IC50 > 10000 nM T55398 CEGF72 44449425 IC50 > 10000 nM T55398 CBA80K 44449426 IC50 = 700 nM T55398 CUY8W6 44449427 IC50 = 2800 nM T55398 CRWG12 44449486 IC50 = 2400 nM T55398 CF0V1N 44449548 IC50 = 3700 nM T55398 C24SWN 44449549 IC50 = 8900 nM T55398 CD6XC0 44449584 IC50 = 4800 nM T55398 C9TR0X 44449617 IC50 = 1000 nM T55398 C3V7EY 44449647 IC50 = 800 nM T55398 CWB60J 44449650 IC50 > 10000 nM T55398 C6DHC9 44450171 IC50 = 7300 nM T55398 C3DQJ6 44450195 IC50 = 7200 nM T55398 CYH6P3 44520205 IC50 = 340 nM T55398 COV31Z 44586245 IC50 = 200 nM T55398 CE3V0Z 44586278 IC50 = 1189 nM T55398 CC5W9J 44586319 IC50 = 456 nM T55398 C8WPI5 44586320 IC50 = 1934 nM T55398 CZI08B 46175395 IC50 = 170 nM T55398 C35UQP 46175482 IC50 = 240 nM T55398 CF0OV6 46175578 IC50 = 1060 nM T55398 CRC37F 46176531 IC50 > 20000 nM T55398 CY3HW5 46224684 IC50 > 10000 nM T55398 COTJ39 46863083 IC50 = 1100 nM T55398 CLS29B 46872626 IC50 > 10000 nM T55398 C1Q8AW 49824621 Ki = 38.5 nM T55398 CAZQ43 51003133 IC50 = 380 nM T55398 CC24GM 52913874 IC50 = 21 nM T55398 CXA03W 52920796 IC50 = 640 nM T55398 CEQN27 52936621 Ki > 1000 nM T55398 C6OTY5 53251320 IC50 = 26000 nM T55398 CE8OY2 53317913 IC50 = 8 nM T55398 C0SWH5 53348216 IC50 > 40000 nM T55398 C8ZRE3 53356518 IC50 > 50000 nM T55398 C8NA4L 53384644 IC50 > 30000 nM T55398 C1XS2J 54760383 IC50 > 10000 nM T55398 C5KR6N 56595558 Ki = 43 nM T55398 COI9U2 56595687 Ki = 420 nM T55398 C2AM6B 56595688 Ki = 1200 nM T55398 CFY2I4 56595689 Ki = 160 nM T55398 CAM8E1 56595690 Ki = 440 nM T55398 CN5EV7 56595691 Ki = 36 nM T55398 C6ET0W 56595693 Ki = 78 nM T55398 CTR10F 56658543 Ki = 340 nM T55398 C9MJG4 56929824 IC50 = 430 nM T55398 C0UDY9 57401151 IC50 = 7500 nM T55398 COY07J 57519810 IC50 <= 5000 nM T55398 C0PA3D 57519811 Ki = 50 nM T55398 CO75VX 58056108 Ki = 1.7 nM T55398 CSN35V 58056134 Ki = 790 nM T55398 C8CG6L 58056265 Ki = 52 nM T55398 CVQ2U4 58056270 Ki = 610 nM T55398 C8GFI0 58056341 Ki = 2 nM T55398 C9MIL7 58450666 IC50 = 1800 nM T55398 C9HUB2 58570982 IC50 = 240 nM T55398 C6BPR2 58985201 IC50 > 30000 nM T55398 CT3EW2 59292007 IC50 > 1000 nM T55398 CP9A8T 59503659 IC50 = 1219 nM T55398 C1MA6J 59503711 IC50 = 1423 nM T55398 CX29EU 59503744 IC50 = 873 nM T55398 CXJ63M 59603829 IC50 = 64 nM T55398 CQEU96 59603842 IC50 = 23 nM T55398 COH62U 60097413 IC50 > 10000 nM T55398 C1MR8Q 60097495 IC50 > 10000 nM T55398 CK6WO0 66552478 IC50 < 10000 nM T55398 CUF20T 66554581 IC50 = 80 nM T55398 CZ92KC 66554752 IC50 = 2100 nM T55398 CF7RQ2 66554923 IC50 = 280 nM T55398 CMS6L3 66554926 IC50 = 180 nM T55398 CU1DM5 66555095 IC50 = 220 nM T55398 CVQW04 66555265 IC50 = 59 nM T55398 C53YWX 66555955 IC50 = 99 nM T55398 CSL0F3 66555956 IC50 = 170 nM T55398 COS5Q9 66555957 IC50 = 44 nM T55398 C7N3DE 66557142 IC50 < 100 nM T55398 C08DXU 66557143 IC50 < 100 nM T55398 COU2C4 66664636 Ki = 8 nM T55398 CV63UL 67240318 IC50 > 10000 nM T55398 C80HMA 68115414 IC50 = 1500 nM T55398 CW23JE 68241353 IC50 = 470 nM T55398 CK9E0Y 68327832 IC50 = 7 nM T55398 CU26SP 68327847 IC50 = 150 nM T55398 CPG75C 68327866 IC50 = 85 nM T55398 CE41YS 68327879 IC50 = 180 nM T55398 CA47UH 68328137 IC50 = 410 nM T55398 C5Z7QJ 68328146 IC50 = 2400 nM T55398 C8OAS6 68328387 IC50 = 27 nM T55398 C3QE9V 68328415 IC50 = 390 nM T55398 CI4HV8 68328491 IC50 = 2 nM T55398 C9HZG1 68328492 IC50 = 40 nM T55398 CC6F8D 68328504 IC50 = 47 nM T55398 C43RXO 68328520 IC50 = 310 nM T55398 CB2OM0 68328789 IC50 = 61 nM T55398 CRM6L5 68357884 IC50 = 5 nM T55398 CZG9X7 68357894 IC50 = 13 nM T55398 C2B1TC 68357902 IC50 = 370 nM T55398 CYI75G 68678653 IC50 = 24400 nM T55398 C5DGR9 69036886 IC50 = 10000 nM T55398 CV0QP3 70947961 Ki = 11 nM T55398 CKT60L 71455860 Ki > 9900 nM T55398 C6T1LM 71506869 IC50 < 50 nM T55398 CE5XR2 71612615 IC50 = 1.8 nM T55398 C5RZ7I 72709739 IC50 = 100 nM T55398 CV3I1N 72943654 IC50 < 100 nM T55398 CIT2V7 72945768 IC50 = 100 nM T55398 CX1UE8 72945946 IC50 = 100 nM T55398 CM94EG 72945952 IC50 > 30000 nM T55398 CZNM96 73053607 IC50 < 100 nM T55398 C25UCH 73053622 IC50 < 100 nM T55398 C1RO3T 73053624 IC50 < 100 nM T55398 CX75YR 73352604 IC50 = 3.981 nM T55398 C8JTD0 73442848 IC50 = 138 nM T55398 CE5CX0 73442898 IC50 = 300 nM T55398 COU3K5 73669498 IC50 = 113 nM T55398 CS2QC6 73669499 IC50 = 204 nM T55398 C7LER5 73669500 IC50 = 3452 nM T55398 C5C4SU 73669664 IC50 = 1140 nM T55398 CF0C4R 73669837 IC50 = 42000 nM T55398 CYO3D1 73669840 IC50 = 2570 nM T55398 C0FH9Y 73670011 IC50 = 1000 nM T55398 C5WLK7 73670169 IC50 = 410 nM T55398 CTG6S3 73670172 IC50 = 333000 nM T55398 C40BHZ 73670173 IC50 = 228000 nM T55398 CJKB83 73670174 IC50 = 11 nM T55398 CF42WG 73670176 IC50 = 4700 nM T55398 C62MPO 73670344 IC50 = 1081000 nM T55398 CW1VG7 73670345 IC50 = 3012000 nM T55398 CJF7Y5 73670346 IC50 = 104 nM T55398 CZU1A0 73670347 IC50 = 24 nM T55398 CCUH57 73670348 IC50 = 16 nM T55398 C82COK 73670350 IC50 = 18 nM T55398 CD23NU 73670513 IC50 = 6000 nM T55398 C1LPW5 73670673 IC50 = 1000 nM T55398 CLO61M 73670847 IC50 = 89 nM T55398 C6T4WZ 73670848 IC50 = 94 nM T55398 CF7TD8 73670850 IC50 = 530 nM T55398 CT3L4F 73670851 IC50 = 932 nM T55398 CN4B8K 75202037 IC50 = 1.5 nM T55398 CFL54M 75204288 IC50 = 1.8 nM T55398 CYJ4C6 76955703 IC50 < 100 nM T55398 CSH9R0 77847460 IC50 < 100 nM T55398 CQ2SU8 78673832 IC50 > 30000 nM T55398 CE0W9R 78673833 IC50 > 30000 nM T55398 C1HW4B 89735655 IC50 = 3000 nM T55398 C89YHN 90134560 IC50 = 5.3 nM T55398 C2CY5A 90154381 IC50 = 3.6 nM T55398 CGTN69 90154630 IC50 = 1.9 nM T55398 C5S0DF 90154917 IC50 = 3.5 nM T55398 CZTM62 90155093 IC50 = 5.6 nM T55398 CAL0O9 90155375 IC50 = 13 nM T55398 CI5GF8 90155577 IC50 = 300 nM T55398 CSC20O 90271946 IC50 = 20 nM T55398 CWA46G 90271957 IC50 < 100 nM T55398 CC1S2P 90272141 IC50 = 71 nM T55398 CM2LJ5 90275527 IC50 = 2400 nM T55398 CNX5V4 91844450 IC50 = 1193000 nM T55398 C0Y8ZK 91933875 IC50 > 1000 nM T55398 CA1K0F 91938073 IC50 = 1.3 nM T55398 CAU45T 91971978 IC50 > 30000 nM T55398 C0YSX8 117826679 IC50 = 4300 nM T55398 CWA8X7 117871492 IC50 = 2197 nM T55398 CI40BM 117871555 IC50 = 3649 nM T55398 CU1V7Y 117871558 IC50 = 187 nM T55398 CQ6E2O 117871721 IC50 > 20000 nM T55398 CTS35E 117871724 IC50 = 3452 nM T55398 CE7X1L 117871750 IC50 = 212 nM T55398 C6MG7L 117871760 IC50 = 730 nM T55398 C0A4XC 117871929 IC50 = 74 nM T55398 CV4B2W 117871992 IC50 = 307 nM T55398 CY60JR 117872182 IC50 = 401 nM T55398 C3VJ0I 117872205 IC50 = 542 nM T55398 CY5JF0 117872250 IC50 = 187 nM T55398 COIM28 117872315 IC50 = 190 nM T55398 C7PM6F 117872316 IC50 = 1100 nM T55398 C63OVX 117872321 IC50 = 653 nM T55398 CT4AZ2 117872334 IC50 = 1100 nM T55398 C6X8VS 117872368 IC50 = 191 nM T55398 CR0JN8 117872469 IC50 = 128 nM T55398 CBOI97 117872492 IC50 = 478 nM T55398 CO6BH7 117872621 IC50 = 1449 nM T55398 CD8J9G 117872890 IC50 = 1605 nM T55398 CQ5S7L 117872990 IC50 = 285 nM T55398 CD6EA9 117873013 IC50 = 2677 nM T55398 C9OA4U 117873033 IC50 = 101 nM T55398 CL6QV4 117873045 IC50 = 261 nM T55398 CDO5I6 117873092 IC50 = 106 nM T55398 CP89EY 117873164 IC50 = 2 nM T55398 C8QB3S 117873179 IC50 = 1582 nM T55398 CWG60S 117873194 IC50 = 2725 nM T55398 CT3B6F 117873210 IC50 = 683 nM T55398 C08YAE 117885624 IC50 = 12 nM T55398 C2V1RC 117885639 IC50 = 830 nM T55398 CS9J3N 117885675 IC50 = 155 nM T55398 CJ8I7U 117885678 IC50 = 12 nM T55398 CK1A0N 117885680 IC50 = 11900 nM T55398 CYP9O7 117885688 IC50 = 12 nM T55398 C4ECT8 117885692 IC50 = 2107 nM T55398 CYN4S1 117885705 IC50 = 3 nM T55398 C2ABD1 117885712 IC50 = 852 nM T55398 CF6UT1 117885715 IC50 = 373 nM T55398 C3VN9K 117885730 IC50 = 7 nM T55398 CZ8P4J 117885751 IC50 = 4 nM T55398 C9R3WU 117885753 IC50 = 6008 nM T55398 C1HND8 117885755 IC50 = 9510 nM T55398 CS72RV 117885758 IC50 = 216 nM T55398 C6Z3NJ 117885766 IC50 = 44 nM T55398 CKU6S4 117885912 IC50 = 8 nM T55398 C1E2DK 118072831 IC50 < 100 nM T55398 C1ZR5E 118173110 IC50 = 33 nM T55398 CV5Q9X 118388894 IC50 = 4381 nM T55398 CT9RU4 118413945 IC50 = 1.3 nM T55398 C36CUE 118414094 IC50 = 0.5 nM T55398 C69QWZ 118414114 IC50 = 29.5 nM T55398 C7J6RO 118414128 IC50 = 4.8 nM T55398 CLWJ18 118414336 IC50 = 7.6 nM T55398 CSQV50 118414357 IC50 = 840 nM T55398 CUJ9O2 118414389 IC50 = 0.1 nM T55398 CF2D3K 118414391 IC50 = 2836 nM T55398 C5XRA6 118414397 IC50 = 23.9 nM T55398 CHL38K 118414437 IC50 = 5.9 nM T55398 CFM20Z 118414536 IC50 = 0.3 nM T55398 CW3IC5 118414671 IC50 = 4.6 nM T55398 C3N5SA 118414693 IC50 = 12.1 nM T55398 CIH2O7 118414733 IC50 = 3.7 nM T55398 C51HAN 118414780 IC50 = 2.7 nM T55398 C0O3SN 118424414 IC50 = 2.4 nM T55398 CUN8Y5 118424424 IC50 = 0.6 nM T55398 COH1T4 118453721 IC50 = 6 nM T55398 CR7DJ0 118453722 IC50 = 55 nM T55398 CK1Z7I 118462026 IC50 = 4 nM T55398 COB6M3 118475320 IC50 = 2 nM T55398 CX2GE1 118475349 IC50 = 250 nM T55398 CZBA29 118641364 IC50 <= 100 nM T55398 CX58DI 118716791 IC50 > 30000 nM T55398 CD9X2B 118716796 IC50 > 30000 nM T55398 C2YJ0O 118716797 IC50 > 30000 nM T55398 CL3UO9 118716798 IC50 > 30000 nM T55398 C71BAM 118716799 IC50 > 30000 nM T55398 CU4EL6 118716806 IC50 > 30000 nM T55398 C5FK7T 118719435 IC50 = 0.36 nM T55398 CA2NJ8 118719437 IC50 = 0.24 nM T55398 CEFG28 118719438 IC50 = 2.8 nM T55398 CL1N2T 118719440 IC50 = 0.32 nM T55398 CCJ0X7 118719442 IC50 = 2.6 nM T55398 CJ2IZ0 118719443 IC50 = 2.2 nM T55398 CIV1H2 118719446 IC50 <= 100 nM T55398 CHT6K9 118728811 Ki > 4000 nM T55398 CUA3Y2 118728812 Ki > 4000 nM T55398 CDQ78G 118728813 Ki > 4000 nM T55398 CZ6XL7 118728814 Ki > 4000 nM T55398 CMO67K 118728815 Ki > 4000 nM T55398 CR2M0Q 118728816 Ki > 4000 nM T55398 C62SCL 118728817 Ki > 4000 nM T55398 CSB30C 118728819 Ki > 4000 nM T55398 CV7XU8 118728820 Ki = 2700 nM T55398 C3J1EX 118728821 Ki > 4000 nM T55398 CIWB78 118728822 Ki > 4000 nM T55398 CP18SE 118728823 Ki = 3300 nM T55398 CM42CA 118728824 Ki > 4000 nM T55398 C9Q7CL 118728825 Ki > 4000 nM T55398 CCR3S0 118728826 Ki > 4000 nM T55398 CNJK97 118729800 IC50 > 20000 nM T55398 C14CYV 118729801 IC50 = 5190 nM T55398 CNP64R 118729802 IC50 > 20000 nM T55398 CP3U7F 118729803 IC50 = 6850 nM T55398 CQ4Z2H 118729804 IC50 > 20000 nM T55398 CQ92UP 118729805 IC50 > 20000 nM T55398 CX9BS1 118729806 IC50 > 20000 nM T55398 C7WFP3 118729807 IC50 > 20000 nM T55398 C3MUB5 118729808 IC50 > 20000 nM T55398 CHDF03 118729809 IC50 > 20000 nM T55398 C6AW4N 118729810 IC50 > 20000 nM T55398 CBWY74 118729811 IC50 = 1140 nM T55398 CN1KS6 118729812 IC50 > 20000 nM T55398 C36BLM 118729813 IC50 = 403000 nM T55398 C4R1EI 121254788 IC50 = 10 nM T55398 C0XU9Y 121255032 IC50 = 7400 nM T55398 CNQ6Z2 121255052 IC50 = 16 nM T55398 CS64MC 121255054 IC50 = 300 nM T55398 CM1W3K 121255069 IC50 = 16 nM T55398 CYDF91 121255074 IC50 = 9 nM T55398 CDQ48W 121255075 IC50 = 19 nM T55398 CZTX30 121256083 IC50 = 12 nM T55398 CJY83B 121258892 IC50 = 17 nM T55398 CTPB07 121262387 IC50 = 32 nM T55398 CUL6H1 121262551 IC50 = 35 nM T55398 C7X1BQ 121493987 IC50 = 38 nM T55398 C30ILY 122180370 IC50 = 690 nM T55398 CK6YL8 122181591 IC50 = 110 nM T55398 CZFT46 122181592 IC50 = 150 nM T55398 COJ93A 122181593 IC50 = 9200 nM T55398 C3EN9U 122181594 IC50 = 2 nM T55398 CWL8R2 122181623 IC50 = 95 nM T55398 CJD5F2 122181624 IC50 = 20 nM T55398 C8C5TR 122181625 IC50 = 8 nM T55398 CT2BY5 122181626 IC50 = 0.3 nM T55398 CYEG26 122181627 IC50 = 14 nM T55398 C06BWF 122181628 IC50 = 6 nM T55398 CEN5P0 122181629 IC50 = 0.8 nM T55398 C6W4PS 122181630 IC50 = 0.3 nM T55398 C1Z0EK 122181631 IC50 = 0.2 nM T55398 CY4HG7 122181632 IC50 = 2 nM T55398 CW74UE 122181633 IC50 = 6 nM T55398 CV87TR 122181634 IC50 = 62 nM T55398 C92TUX 122181635 IC50 = 160 nM T55398 CSD5U0 122181636 IC50 = 480 nM T55398 CC3FS4 122181637 IC50 = 21 nM T55398 CD83YT 122181638 IC50 = 4 nM T55398 CVQ7H5 122181639 IC50 = 10 nM T55398 CTD2I5 122181640 IC50 = 1 nM T55398 CKJU62 122181641 IC50 = 23 nM T55398 CMQ2R0 122181642 IC50 = 13 nM T55398 C4WZR2 122181643 IC50 = 3 nM T55398 CF2LI0 122181644 IC50 = 3 nM T55398 CMZ95X 122181645 IC50 = 1 nM T55398 CFU63N 122181674 IC50 = 0.5 nM T55398 CF7OC2 122181675 IC50 = 0.5 nM T55398 C76RQM 122181676 IC50 = 6 nM T55398 C8D3JG 122184715 IC50 = 11 nM T55398 C0BLW3 122184716 IC50 = 647 nM T55398 CAQ71B 122191866 IC50 = 470 nM T55398 CO6S2E 122196062 IC50 = 40 nM T55398 C8R7FJ 122196063 IC50 = 5 nM T55398 CJA40H 122196064 IC50 = 1 nM T55398 CV85FQ 122196065 IC50 = 10 nM T55398 CBW67H 122196066 IC50 = 1 nM T55398 C7W5QA 122196067 IC50 = 0.2 nM T55398 CS6AP9 122196068 IC50 = 38 nM T55398 CJO8V9 122196168 IC50 = 3 nM T55398 CVI2P6 122196169 IC50 < 0.5 nM T55398 CO72HB 122196170 IC50 = 2 nM T55398 CA6BO3 122196171 IC50 = 1 nM T55398 CU2XL4 122196172 IC50 = 0.8 nM T55398 CZ3W8X 122196173 IC50 < 0.5 nM T55398 CB21TD 122196174 IC50 = 24 nM T55398 C51YFU 122196175 IC50 = 0.9 nM T55398 CX07CU 122196176 IC50 = 0.4 nM T55398 C2HLK9 122196177 IC50 = 0.2 nM T55398 C84DQM 122196178 IC50 = 0.7 nM T55398 C0DO3U 122196179 IC50 < 0.5 nM T55398 CYMK98 122196180 IC50 = 1 nM T55398 CQ1OM7 122196181 IC50 = 1 nM T55398 CLFH30 122196246 IC50 = 7 nM T55398 C5Z2FM 122196247 IC50 = 25 nM T55398 CTX0M5 122196248 IC50 = 12 nM T55398 C43LHP 122196249 IC50 = 0.4 nM T55398 C6QZE1 123917405 IC50 = 2400 nM T55398 CZEV34 125479776 IC50 = 1200 nM T55398 CR3A1O 125495464 IC50 = 15 nM T55398 CGU28T 126573669 IC50 = 121 nM T55398 C2T8ZA 126573681 IC50 = 146 nM T55398 C4S5LR 126622195 IC50 = 0.2 nM T55398 CH4C5O 126961337 IC50 = 58 nM T55398 CAGL14 126970816 IC50 = 71.9 nM T55398 C31ZLG 127034634 Ki = 7.8 nM T55398 CX3YO4 127034635 Ki = 11 nM T55398 CUS38N 127034643 IC50 = 150 nM T55398 C1C4UV 127034834 Ki = 3.8 nM T55398 CZ7H8F 127035289 Ki = 1.6 nM T55398 CZD87E 127037084 IC50 = 465 nM T55398 CB9Z0V 127038973 IC50 = 234 nM T55398 C1KH4L 129284027 Ki = 30 nM T55398 C6RGX5 129284078 Ki = 2.1 nM T55398 C9VL8H 129284112 Ki = 7.4 nM T55398 CWF79O 129284190 Ki = 14 nM T55398 CBJ6X9 129284195 IC50 = 0.38 nM T55398 C3VK4I 129284254 Ki = 7.3 nM T55398 C4VS8P 129284274 Ki = 35 nM T55398 CK2IL4 129284334 IC50 = 0.19 nM T55398 C96LDG 129284345 Ki = 5.1 nM T55398 CN8WZ2 129284370 Ki = 80 nM T55398 C8VNP1 129284385 IC50 = 7.2 nM T55398 CWA5R2 129284395 Ki = 6.6 nM T55398 CR2YV6 129284442 IC50 = 3.6 nM T55398 C4MG6I 129284483 Ki = 1.1 nM T55398 C9W4CS 129284507 Ki = 6.1 nM T55398 CR94JT 129284517 Ki = 3.5 nM T55398 CF19RT 129284574 Ki = 15 nM T55398 CM2J9U 129284575 Ki = 13 nM T55398 C49BMA 129284616 Ki = 6.1 nM T55398 CO4QV7 129284658 Ki = 1.5 nM T55398 C43SGU 129284679 Ki = 31 nM T55398 CS71NJ 129284701 Ki = 34 nM T55398 CV25CZ 129284859 Ki = 3.2 nM T55398 CM23FX 129297015 Ki = 12 nM T55398 CQO83S 129297033 Ki = 10 nM T55398 C0Z5NP 129297518 Ki = 5.8 nM T55398 C2FU6N 129297531 IC50 = 1.2 nM T55398 CFSC56 129297811 Ki = 3.2 nM T55398 C4NG3W 129298165 IC50 = 0.16 nM T55398 CUOX69 129298210 IC50 = 0.081 nM T55398 CTA06R 129298213 IC50 = 0.32 nM T55398 C96KMC 129298275 Ki = 6.5 nM T55398 C8MXQ4 130274633 IC50 = 7 nM T55398 CK4N0V 130274681 IC50 = 122 nM T55398 C45OHZ 130275697 IC50 = 3 nM T55398 C18QMF 130275783 IC50 = 3 nM T55398 C3WG8E 130276452 IC50 = 8 nM T55398 C9WK5I 130276470 IC50 = 17 nM T55398 CXTZ19 131704459 IC50 = 10 nM T55398 C25WQI 131704460 IC50 > 10000 nM T55398 CY70JL 131839618 IC50 = 6 nM T55398 C4Z5MQ 131839619 IC50 = 5 nM T55398 C2W8TC 131839620 IC50 = 42 nM T55398 C0M7PT 131839621 IC50 = 2 nM T55398 CNF79T 133107904 IC50 = 4 nM T55398 CB0C4Y 133107905 IC50 = 69 nM T55398 CJ43BV 133107906 IC50 = 21.38 nM T55398 C2AN7T 134611886 IC50 > 100000 nM T55398 CY4D8I 135566504 Ki > 1000 nM T55398 C7PJ6X 135566704 IC50 > 30000 nM T55398 C6DP4U 135567024 IC50 = 25 nM T55398 CX3UR8 135567025 IC50 = 19 nM T55398 CPV59N 135685787 Ki = 1500 nM T55398 CG3UZ1 135927974 Ki > 1000 nM T55398 CF1PS8 135934877 Ki = 690 nM T55398 CTRL59 135976660 Ki = 1100 nM T55398 CU0SZ4 136074298 IC50 < 100 nM T55398 CDMS84 136074299 IC50 < 100 nM T55398 CSOR07 136074300 IC50 = 14 nM T55398 CQ84IZ 136180335 Ki > 4000 nM T55398 COLR97 136272332 IC50 = 1487 nM T55398 CS9Z2N 136272346 IC50 = 1688 nM T55398 CX48MU 136272376 IC50 = 11 nM T55398 CYUF15 136272377 IC50 = 78 nM T55398 CL6S3R 136272378 IC50 = 43 nM T55398 C6T7AE 136272379 IC50 = 135 nM T55398 C7Y1QZ 136272387 IC50 = 43 nM T55398 C2V7QH 136272388 IC50 = 27 nM T55398 CN49DR 136272389 IC50 = 490 nM T55398 C7XY1B 136272390 IC50 = 67 nM T55398 COQ3V4 136504460 IC50 = 972 nM T55398 CVPE08 136504461 IC50 = 2429 nM T55398 CB0M7Z 136504482 IC50 = 454 nM T55398 C7ZF1S 136508720 IC50 = 79 nM T55398 CY1Q8P 136508752 IC50 = 85 nM T55398 C5K8ED 136932639 IC50 = 565 nM T55398 C9DF2X 136932640 IC50 = 580 nM T55398 C9IS5M 136983815 IC50 = 121 nM T55398 C9V3KL 136983853 IC50 = 258 nM T55398 CHT7X2 136983871 IC50 = 352 nM T55398 C24BNM 136983876 IC50 = 635 nM T55398 C39FNY 136983894 IC50 = 36 nM T55398 CWL74T 136983918 IC50 = 354 nM T55398 CSJI86 136983949 IC50 = 620 nM T55398 C3R0PB 136984063 IC50 = 450 nM T55398 C5KN9F 136984064 IC50 = 100 nM T55398 CH3M4B 137083628 IC50 > 30000 nM T55398 CJA07O 137083629 IC50 > 30000 nM T55398 C9F8PX 137083630 IC50 = 579 nM T55398 C96CJQ 137348875 IC50 = 360 nM T55398 C8GD6Y 137367179 IC50 = 0.47 nM T55398 CT2FE0 137367190 IC50 = 0.11 nM T55398 C52UFH 137367200 Ki = 210 nM T55398 C3PBN7 137367378 IC50 = 0.026 nM T55398 CZ4VW3 137631374 IC50 = 21 nM T55398 C0U4AO 137631449 IC50 = 10 nM T55398 CN32XA 137631833 IC50 = 82 nM T55398 C90ELI 137631990 IC50 = 730 nM T55398 CSVD52 137632007 IC50 = 20 nM T55398 C0OWI4 137632095 IC50 = 3 nM T55398 CQU8G7 137632864 IC50 = 33 nM T55398 CZH08K 137633516 IC50 = 180 nM T55398 CC9IU4 137634304 IC50 = 5 nM T55398 CYEO71 137634466 IC50 = 5 nM T55398 CQR3H5 137634670 IC50 = 140 nM T55398 CXG74K 137635345 IC50 = 50 nM T55398 CY6TH8 137635761 IC50 = 4.571 nM T55398 CJE35M 137636090 IC50 = 20 nM T55398 C8Z9VW 137637011 IC50 = 3 nM T55398 C1KWC2 137637354 IC50 = 99 nM T55398 CPEI56 137637758 IC50 = 16 nM T55398 CE8AB3 137639678 IC50 = 400 nM T55398 CB6GD5 137639959 IC50 = 47 nM T55398 CB0JI5 137640711 IC50 = 2000 nM T55398 CO1MS6 137641896 IC50 = 14600 nM T55398 CY9QE7 137642189 IC50 = 4.786 nM T55398 CA9DE5 137642519 IC50 = 390 nM T55398 CP6K0U 137642747 IC50 = 120 nM T55398 C47KFJ 137642928 IC50 = 4 nM T55398 C1BK8H 137643835 IC50 = 9 nM T55398 CBA59R 137644862 IC50 = 1300 nM T55398 CP74MV 137644945 IC50 = 75 nM T55398 C7KHW3 137645090 IC50 = 410 nM T55398 CXIN67 137645231 IC50 = 58 nM T55398 C0GYU1 137646905 IC50 = 8 nM T55398 CGU2E5 137648767 IC50 = 840 nM T55398 CQHO93 137649163 IC50 = 3 nM T55398 CBY15N 137649190 IC50 = 56 nM T55398 CX8N6D 137650526 IC50 = 13 nM T55398 C98RIA 137651604 IC50 = 270 nM T55398 C0RUL8 137651621 IC50 = 10 nM T55398 CFX6Y3 137651671 IC50 = 13 nM T55398 C5NUY0 137651713 IC50 = 25 nM T55398 C7BJN4 137652293 IC50 = 170 nM T55398 C5CKI4 137652730 IC50 = 64 nM T55398 CAFG38 137653032 IC50 = 630.96 nM T55398 C8UGS4 137653281 IC50 = 50 nM T55398 CQT9B3 137653599 IC50 = 13 nM T55398 CS6RE8 137654629 IC50 = 50 nM T55398 CNIX25 137655529 IC50 = 1600 nM T55398 C27SVK 137656133 IC50 = 11 nM T55398 CR8Z9G 137656476 IC50 = 2087 nM T55398 CQ0GX8 137657147 IC50 = 40 nM T55398 CLW29O 137657406 IC50 = 9000 nM T55398 C49DOZ 137657630 IC50 = 19 nM T55398 CXS2U8 137658175 IC50 = 34 nM T55398 CO6XD2 137658443 IC50 = 22 nM T55398 CU0ST8 137659008 IC50 = 130 nM T55398 C6Z8YN 137659188 IC50 = 70 nM T55398 CB1XR5 137659870 IC50 = 4 nM T55398 CMZ36T 137659999 IC50 = 730 nM T55398 CK1B4W 137660846 IC50 = 6 nM T55398 CM23OE 137661767 IC50 = 44 nM T55398 CJ0G3C 138376590 Ki = 1.8 nM T55398 CX64WE 138620530 IC50 < 30 nM T55398 C2LHE0 138620547 IC50 < 30 nM T55398 CA63ML 138620560 IC50 < 30 nM T55398 CR0Y8I 138656676 IC50 < 30 nM T55398 CA1I4Y 138656977 IC50 < 30 nM T55398 C72APW 138727769 IC50 = 97.72 nM T55398 C5J2WV 138728749 IC50 = 94 nM T55398 CVU63L 139582016 IC50 = 37 nM T55398 C8PH9S 139582017 IC50 = 4 nM T55398 C45PVO 142501440 Ki = 22 nM T55398 CU12BZ 142501542 IC50 = 0.1 nM T55398 CV1KM9 145979754 IC50 = 77.62 nM T55398 CX05ZN 145979845 IC50 = 22 nM T55398 CY9X5Q 145979885 IC50 = 1190 nM T55398 C9N2XW 145980788 IC50 = 19.5 nM T55398 CNQ67H 145987089 IC50 = 207 nM T55398 C1N9LZ 145987466 IC50 = 446 nM T55398 C9O6WH 145987619 IC50 = 1530 nM T55398 C4QX5P 145987677 IC50 = 44.67 nM T55398 CYS4V9 145990152 IC50 = 234.42 nM T55398 C3T6XI 145991666 IC50 = 1770 nM T55398 CEL5Y6 145991871 IC50 = 738 nM T55398 CP15XW 145992518 IC50 = 33 nM T55398 CSHF19 145992913 IC50 = 602.56 nM T55398 C1N8CA 145993210 IC50 = 671 nM T55398 C12VLN 145993338 IC50 = 87.1 nM T55398 CE9PV2 145993467 IC50 > 10000 nM T55398 CT74QG 145993512 IC50 = 4073.8 nM T55398 C2B4VW 145993656 IC50 = 42 nM T55398 C5H2WU 145993757 IC50 = 16 nM T55398 CHT23F 145993921 IC50 = 804 nM T55398 C6PK4L 146483027 IC50 = 0.078 nM T55398 CMZ4J3 155510495 IC50 < 30 nM T55398 CHX57D 155511560 Ki = 95 nM T55398 CKB64L 155512869 IC50 = 69 nM T55398 C2MD1Q 155513187 IC50 > 10000 nM T55398 C93SNT 155514207 IC50 = 1 nM T55398 C17BHJ 155516763 IC50 = 0.022 nM T55398 C08VAM 155517957 IC50 = 2.5 nM T55398 C8UI7G 155520013 IC50 = 0.29 nM T55398 CCL0S9 155520435 IC50 = 0.099 nM T55398 C7YSD8 155522882 IC50 > 5000 nM T55398 C70GEI 155525183 IC50 > 5000 nM T55398 CWP05R 155527255 Ki = 1.7 nM T55398 CE2YX6 155527737 Ki = 290 nM T55398 CSGV07 155529499 Ki > 8400 nM T55398 CA83QP 155529897 IC50 > 5000 nM T55398 CGDE18 155530136 IC50 > 5000 nM T55398 CSJB85 155530835 Ki = 0.5 nM T55398 CWU8N1 155535119 IC50 = 38 nM T55398 CL5F3C 155537218 Ki = 0.5 nM T55398 CG4LQ2 155539650 Ki = 1.2 nM T55398 C29FDV 155542370 IC50 = 9 nM T55398 C8NOD0 155544794 Ki > 30000 nM T55398 CX9FM8 155548286 IC50 = 2.1 nM T55398 CSJ72Y 155549539 IC50 = 6 nM T55398 CR79JM 155549965 IC50 = 1 nM T55398 CN6O2U 155552158 IC50 > 5000 nM T55398 CM8O9G 155552851 Ki = 170 nM T55398 CWO25P 155555362 Ki = 26 nM T55398 C4Y6BV 155556454 Ki = 6.7 nM T55398 C0WUZ4 155556888 IC50 = 5 nM T55398 C8NMG3 155558108 IC50 > 5000 nM T55398 CWJ08R 155560232 Ki = 0.8 nM T55398 C4IP2Y 155561648 IC50 = 17 nM T55398 C0EBX7 155561943 IC50 = 279 nM T55398 C3D2GP 155562155 IC50 = 21 nM T55398 D00ERW 44444843 Ki > 9921 nM T55398 D00HVA 11624601 Ki > 9900 nM T55398 D02JIL 3572750 IC50 = 4000 nM T55398 D04CFM 86343751 Ki = 1 nM T55398 D04ZIV 58056241 IC50 = 1 nM T55398 D06HVH 54613583 IC50 > 10000 nM T55398 D06WGX 9549184 IC50 > 25000 nM T55398 D09JUD 44449334 IC50 = 20 nM T55398 D0I2FZ 11983295 IC50 = 200 nM T55398 D0J3LR 11634725 Ki > 4000 nM T55398 D0J8VR 25169383 IC50 = 1 nM T55398 D0LY5S 2635761 IC50 = 13600 nM T55398 D0ME9B 46868971 IC50 = 1800 nM T55398 D0Q3NG 11715520 Ki > 9900 nM T55398 D0S7IE 11658882 Ki > 9900 nM T55398 D0T2NE 58056092 IC50 = 8 nM T55398 D0Y2ZC 68115559 IC50 = 7.5 nM T66505 D03EDQ 24776445 IC50 = 5.1 nM T66505 D03LWG 53235510 Ki = 46.5 nM T66505 D04MXN 56846693 Ki = 187.8 nM T66505 D08FDX 24901704 Ki = 41.7 nM T66505 D09BNZ 24775005 Ki = 6 nM T66505 D09UMN 45100669 IC50 < 100 nM T66505 D0D1GF 42642645 Ki = 59.7 nM T66505 D0GD4Q 25027363 IC50 = 1.4 nM T66505 D0M9QZ 11485656 Ki = 87.6 nM T66505 C5V3DJ 1048811 Ki = 50.4 nM T66505 CBVR03 1139102 IC50 = 281 nM T66505 C5W4RP 1300425 IC50 = 89 nM T66505 C0MHW2 2270563 IC50 = 109 nM T66505 C80TKI 2952255 IC50 = 4.4 nM T66505 CFWS91 2953198 IC50 = 91 nM T66505 C1FQR3 3537781 IC50 = 13 nM T66505 CVOH96 3591787 IC50 > 2500 nM T66505 C0LY1H 4269048 Ki = 168.1 nM T66505 CB9I0U 5284329 IC50 = 1500 nM T66505 CK73QZ 6405276 IC50 = 13 nM T66505 CEA26I 6407374 IC50 = 19 nM T66505 C8UB6G 6878030 IC50 = 4.74 nM T66505 CR4Z0H 8440567 IC50 = 1860 nM T66505 C2MJB3 9869236 IC50 = 3420 nM T66505 CLH27B 10392802 IC50 = 140 nM T66505 C1IZR8 10951208 IC50 = 120 nM T66505 CL4BI2 11762419 IC50 = 7520 nM T66505 C2JYM1 18526613 IC50 = 1243 nM T66505 CKU1F2 20875737 IC50 > 5000 nM T66505 C4C9WL 22291085 IC50 = 450 nM T66505 CK6P2Z 24797888 IC50 = 170 nM T66505 CY69VQ 24797889 IC50 = 10 nM T66505 C16WVQ 24797980 IC50 = 240 nM T66505 CZ3EV7 24798071 IC50 = 120 nM T66505 CKYJ26 24905375 IC50 = 8 nM T66505 CN97YF 25065064 IC50 = 724 nM T66505 CEJT74 25065069 IC50 = 2261 nM T66505 CV3R7X 25065678 IC50 = 34 nM T66505 C24YFH 25065681 IC50 = 82 nM T66505 C0HPL9 25065893 IC50 = 185 nM T66505 CJ68BR 25065894 IC50 = 196 nM T66505 CC90KI 25066322 IC50 > 5000 nM T66505 C5UGO6 25066518 IC50 = 112 nM T66505 CGI08J 25066520 IC50 = 95 nM T66505 CYL6V4 25067132 IC50 = 391 nM T66505 CEA5R6 25181471 IC50 < 6 nM T66505 CVPH81 25210551 IC50 = 2700 nM T66505 CI6VC1 25211577 IC50 = 7 nM T66505 CUWT70 25211578 IC50 = 7 nM T66505 CJPE39 25211677 IC50 = 770 nM T66505 CJ0C6Z 25224531 IC50 = 16 nM T66505 C2GBS5 25224707 IC50 = 66 nM T66505 CNX9T4 25226761 IC50 = 1 nM T66505 CUL3B0 25226762 IC50 = 5.8 nM T66505 CCP60F 25226764 IC50 = 12 nM T66505 CC7GX8 25253556 IC50 < 12 nM T66505 C7WZY2 25255940 IC50 = 2.8 nM T66505 CR63VO 44186114 IC50 > 5000 nM T66505 CAU96H 44186115 IC50 = 59 nM T66505 C8I5FZ 44186181 IC50 = 217 nM T66505 CB7K3J 44186182 IC50 > 5000 nM T66505 CBQD07 44186183 IC50 > 5000 nM T66505 C8OLT2 44186184 IC50 = 401 nM T66505 C2EIF1 44186185 IC50 = 230 nM T66505 C9ROY5 44186310 IC50 = 306 nM T66505 CM4SK2 44186312 IC50 = 654 nM T66505 CB5US1 44186313 IC50 = 15 nM T66505 CGR97M 44186314 IC50 = 484 nM T66505 CQ58TU 44186375 IC50 = 67 nM T66505 CJD40V 44186376 IC50 = 21 nM T66505 C3QDF2 44186378 IC50 = 70 nM T66505 CS96ZI 44186429 IC50 = 103 nM T66505 C0L4ES 44186430 IC50 = 25 nM T66505 C1PTH6 44186431 IC50 = 2929 nM T66505 CM8H5Z 44186480 IC50 = 34 nM T66505 C31RVS 44186482 IC50 = 17 nM T66505 C8Z1DQ 44186485 IC50 > 5000 nM T66505 CQT23O 44186526 IC50 > 5000 nM T66505 C6BD5U 44250034 IC50 = 5 nM T66505 CZTH83 44250105 IC50 = 40 nM T66505 C8H9TQ 44395035 IC50 = 3200 nM T66505 C0T2GL 44395101 IC50 = 1100 nM T66505 CY9R4E 44395109 IC50 = 450 nM T66505 C0MT1L 44395257 IC50 > 3000 nM T66505 CF9IW1 44412191 IC50 = 78.4 nM T66505 C1NF9R 44463317 IC50 = 90 nM T66505 CT14KB 44464376 IC50 = 190 nM T66505 CE7J2C 44464620 IC50 = 107 nM T66505 CYJ02G 44464875 IC50 = 80 nM T66505 CYLN29 44517800 IC50 = 31 nM T66505 C3O7TI 44548374 IC50 = 44 nM T66505 C7CJM3 44548378 IC50 = 93 nM T66505 CY9M7W 44549004 IC50 = 40 nM T66505 CRT70E 44591268 IC50 = 30 nM T66505 CQE8H0 44591290 IC50 = 790 nM T66505 C7ZX3O 44591292 IC50 = 1150 nM T66505 C5VUK4 44591325 IC50 = 14 nM T66505 CF1E9T 44591326 IC50 = 340 nM T66505 CVB19K 44591344 IC50 = 32 nM T66505 CMR54E 44591345 IC50 = 55 nM T66505 CPW59G 44591346 IC50 = 210 nM T66505 CO31UZ 44591347 IC50 = 130 nM T66505 CZ2C0W 44610687 IC50 = 380 nM T66505 C4U9EN 44628220 IC50 = 3400 nM T66505 CKM92Y 44628222 IC50 = 2200 nM T66505 CO72KB 44628287 IC50 = 1100 nM T66505 C0YM5V 44628288 IC50 = 1500 nM T66505 CV9A3W 44628450 IC50 = 1200 nM T66505 CMA16F 44628452 IC50 = 1500 nM T66505 CAW8Y9 44628525 IC50 = 320 nM T66505 CK0G2O 44628528 IC50 = 1800 nM T66505 CZY63O 44628618 IC50 = 420 nM T66505 C62FGB 44628620 IC50 = 1300 nM T66505 CPG83O 44628898 IC50 > 2500 nM T66505 CS37ZL 44629065 IC50 = 790 nM T66505 CEX0I1 44629066 IC50 = 1000 nM T66505 CVS96Z 44629067 IC50 = 280 nM T66505 CL9N4Z 44629071 IC50 = 520 nM T66505 CER8Q0 44629155 IC50 = 470 nM T66505 C8XGK2 44629232 IC50 = 510 nM T66505 CDQ47G 44629236 IC50 = 700 nM T66505 CGW6U0 44629295 IC50 = 750 nM T66505 CX1QC4 44629366 IC50 > 2500 nM T66505 CE6B2G 45267515 IC50 = 130 nM T66505 CF8VX0 45267523 IC50 > 10000 nM T66505 CUW4Z0 45267528 IC50 = 70 nM T66505 C0Z3MB 45267540 IC50 = 1800 nM T66505 CUM1G5 45268389 IC50 = 10000 nM T66505 CYU5Q0 45268404 IC50 = 310 nM T66505 CC7H9M 45268408 IC50 = 200 nM T66505 C9VCH6 45268412 IC50 = 100 nM T66505 CS90AD 45269254 IC50 = 3000 nM T66505 CHCB29 45269261 IC50 = 900 nM T66505 CH3NB9 45269264 IC50 = 950 nM T66505 CD0FN3 45270098 IC50 = 1200 nM T66505 CI16LK 45270102 IC50 = 360 nM T66505 CKNH75 45270116 IC50 = 130 nM T66505 CH2F3N 45270117 IC50 > 25000 nM T66505 CRO2M3 45270118 IC50 = 6300 nM T66505 C3PTM6 45270935 IC50 = 720 nM T66505 CN2F0B 45270940 IC50 = 900 nM T66505 CI95MH 45270943 IC50 = 200 nM T66505 C29UPR 45270944 IC50 = 120 nM T66505 CDV71Y 45270956 IC50 = 1400 nM T66505 CGYD64 45271780 IC50 = 10000 nM T66505 CQ9K4Y 45271789 IC50 = 1300 nM T66505 CF12YU 45271790 IC50 = 1200 nM T66505 C2P1MF 45272645 IC50 = 10000 nM T66505 CL1S7X 45272649 IC50 = 10000 nM T66505 CL91PA 45272656 IC50 = 680 nM T66505 CGO7B5 45272667 IC50 > 10000 nM T66505 CB6S7D 45272668 IC50 = 1830 nM T66505 C3C1DS 45273570 IC50 = 330 nM T66505 CES8O2 45273586 IC50 = 150 nM T66505 C1B4AO 45273591 IC50 = 4500 nM T66505 CIQ7M3 45273599 IC50 = 340 nM T66505 CK7XM8 46871826 IC50 = 5.3 nM T66505 CP87LJ 46871827 IC50 = 2.2 nM T66505 CT8FV6 46890873 IC50 = 9.5 nM T66505 CXY13W 46890935 IC50 = 13 nM T66505 C1CIG5 46890990 IC50 = 5.3 nM T66505 CVBK65 46890991 IC50 = 17.3 nM T66505 CIZ8O7 46890992 IC50 = 5.2 nM T66505 C4GR0D 46891044 IC50 = 15 nM T66505 CMT7B2 46891045 IC50 = 10.8 nM T66505 CH1K0L 46891046 IC50 = 20 nM T66505 CY0T2V 46891103 IC50 = 212 nM T66505 CY0A3H 46891104 IC50 = 15 nM T66505 CRW3N1 46891105 IC50 = 20.3 nM T66505 C1V4PY 46891106 IC50 = 110 nM T66505 C2JRG0 46891162 IC50 = 213 nM T66505 C1PC7R 46891163 IC50 = 96 nM T66505 CK6RY3 46891164 IC50 = 3.2 nM T66505 CE46PC 46891165 IC50 = 7 nM T66505 C1JFY6 46891197 IC50 = 11.8 nM T66505 CHQ06G 46891198 IC50 = 3.6 nM T66505 CAYC57 46891199 IC50 = 0.7 nM T66505 CLD87G 46891200 IC50 = 0.4 nM T66505 CVK3A7 46891245 IC50 = 2.3 nM T66505 CQCN85 46891246 IC50 = 7.3 nM T66505 C0NF6E 46891247 IC50 = 10.1 nM T66505 CY89AF 46891248 IC50 = 2.7 nM T66505 C7D9UV 46891298 IC50 = 3.1 nM T66505 CH03ZS 46891299 IC50 = 5.2 nM T66505 CV6MN7 46891300 IC50 = 2340 nM T66505 C59RFZ 46891346 IC50 = 2700 nM T66505 C24DXJ 49840814 IC50 = 4 nM T66505 C2O7ZC 49862152 IC50 = 1870 nM T66505 C9AQO8 49862153 IC50 = 1690 nM T66505 C0AY1M 49862154 IC50 = 20 nM T66505 CSR2H4 49862176 IC50 = 12 nM T66505 CPNL82 49862194 IC50 > 5000 nM T66505 CN0V7S 49862195 IC50 > 5000 nM T66505 CFNZ30 49862196 IC50 = 333 nM T66505 C06TVH 49862197 IC50 = 105 nM T66505 C7H2NL 49862220 IC50 = 19 nM T66505 C0U7CJ 49862221 IC50 = 21 nM T66505 CIUH50 49862222 IC50 > 1000 nM T66505 CZ8GI9 49862236 IC50 = 64.7 nM T66505 C6OQV2 49862237 IC50 = 40.8 nM T66505 C6IW4Q 49862238 IC50 = 8.27 nM T66505 CP1YK8 49862269 IC50 = 3.3 nM T66505 C4HRQ3 49862270 IC50 = 4.8 nM T66505 CCL25Y 49862311 IC50 = 25 nM T66505 C16VMC 49862312 IC50 = 79 nM T66505 C7H5LT 49862313 IC50 = 57 nM T66505 C1J9KL 49862314 IC50 = 8.7 nM T66505 CI0Q6T 49862371 IC50 = 8 nM T66505 C8GS6K 49862372 IC50 > 1000 nM T66505 CB10HZ 49862373 IC50 > 1000 nM T66505 C4FYZ5 49862424 IC50 > 1000 nM T66505 C3QF1T 50768213 IC50 > 2500 nM T66505 CXN52T 50835422 IC50 = 63 nM T66505 CRZL59 53361076 IC50 = 13 nM T66505 C0CE7M 53387030 IC50 = 13 nM T66505 C1RHF7 53387681 IC50 = 5 nM T66505 CTY6C4 53484000 IC50 = 7.2 nM T66505 C13WTO 56658050 IC50 = 46 nM T66505 C8GZD4 56658051 IC50 = 2600 nM T66505 CT62BA 56658169 IC50 = 230 nM T66505 CJDL15 56658170 IC50 = 2000 nM T66505 C30TCQ 56658188 IC50 = 6.4 nM T66505 CV68SR 56658189 IC50 = 48 nM T66505 CL38IE 56658549 IC50 = 180 nM T66505 C4U7WK 56658550 IC50 = 4700 nM T66505 C0G4XL 56658551 IC50 > 2500 nM T66505 C7MBL0 56658552 IC50 > 2500 nM T66505 C75ITF 56658553 IC50 > 2500 nM T66505 C1SH5E 56658575 IC50 = 480 nM T66505 CV2EY4 56658696 IC50 > 2500 nM T66505 CA9KM7 56658697 IC50 = 480 nM T66505 CV6T7E 56658698 IC50 > 2500 nM T66505 CW72LF 56658699 IC50 > 2500 nM T66505 CCA76B 56661560 IC50 = 46 nM T66505 C4H3VZ 56661561 IC50 = 340 nM T66505 CRI23C 56661562 IC50 = 64 nM T66505 C43ICJ 56661679 IC50 = 72 nM T66505 C8D9PR 56662002 IC50 = 15000 nM T66505 C35SAR 56662003 IC50 = 620 nM T66505 CG2U1T 56662004 IC50 = 1000 nM T66505 C9BNK7 56662005 IC50 = 1900 nM T66505 CY26QZ 56662006 IC50 > 2500 nM T66505 CQ41MY 56662174 IC50 = 110 nM T66505 CB4W0O 56662175 IC50 > 2500 nM T66505 CVSD83 56662176 IC50 = 670 nM T66505 C8E5BX 56662793 IC50 = 18 nM T66505 C3PKE1 56663266 IC50 = 3000 nM T66505 CM2O8C 56664980 IC50 = 330 nM T66505 C92THJ 56664981 IC50 = 380 nM T66505 C1ME2L 56665113 IC50 = 37 nM T66505 CAY4Z3 56665494 IC50 = 640 nM T66505 CT9O7X 56665495 IC50 = 6000 nM T66505 CWCK98 56665496 IC50 > 2500 nM T66505 C41XMQ 56665497 IC50 = 2200 nM T66505 CG75HU 56665498 IC50 > 2500 nM T66505 CKA36R 56665499 IC50 > 2500 nM T66505 CKB71O 56665632 IC50 > 2500 nM T66505 CMJ13X 56666699 IC50 = 4600 nM T66505 CX4IC9 56668414 IC50 = 200 nM T66505 CX8Q5Y 56668540 IC50 = 13000 nM T66505 CUFX01 56668541 IC50 = 240 nM T66505 CF7LR5 56668542 IC50 = 32 nM T66505 CI4Q1R 56668557 IC50 = 49 nM T66505 C6KVX4 56668558 IC50 = 27 nM T66505 C2DR5K 56668559 IC50 = 27 nM T66505 CU19OY 56668560 IC50 = 93 nM T66505 CG6JS7 56668711 IC50 = 810 nM T66505 C8W4QB 56668923 IC50 > 2500 nM T66505 CP9U0G 56668924 IC50 = 1000 nM T66505 C02GYK 56668936 IC50 = 45 nM T66505 CMQS94 56669087 IC50 = 1900 nM T66505 C5W8BE 56669674 IC50 = 140 nM T66505 CQJ72G 56669675 IC50 = 100 nM T66505 C51HRV 56669676 IC50 = 15 nM T66505 CR9IJ2 56669677 IC50 = 21 nM T66505 C3IE7S 56671926 IC50 = 530 nM T66505 CYOA69 56671927 IC50 = 390 nM T66505 C5RFI6 56671928 IC50 = 19 nM T66505 CTL7J0 56671929 IC50 = 8 nM T66505 C68YBP 56672043 IC50 = 4900 nM T66505 C4XK3V 56672054 IC50 = 14 nM T66505 CVCW54 56672401 IC50 > 2500 nM T66505 C8CMQ3 56672402 IC50 = 1100 nM T66505 C67POD 56672403 IC50 > 2500 nM T66505 C60FCS 56672404 IC50 > 2500 nM T66505 CK8Y7L 56672544 IC50 = 490 nM T66505 CY8Q6Z 56672545 IC50 = 750 nM T66505 C9O6JQ 56672546 IC50 = 2900 nM T66505 CP0J8E 56672547 IC50 = 1300 nM T66505 COI7L2 56673182 IC50 = 1200 nM T66505 CI9QV5 56675303 IC50 = 790 nM T66505 CO4ND2 56675304 IC50 = 510 nM T66505 CKXE70 56675305 IC50 = 2700 nM T66505 CTE98L 56675306 IC50 = 17000 nM T66505 C5O7WK 56675307 IC50 = 290 nM T66505 CWI58T 56675308 IC50 = 15 nM T66505 CI06FK 56675419 IC50 = 6900 nM T66505 CJEA89 56675420 IC50 = 290 nM T66505 CK57CI 56675440 IC50 = 28 nM T66505 CM5UH2 56675441 IC50 = 33 nM T66505 CY6UA5 56675678 IC50 > 2500 nM T66505 C9C8FG 56675786 IC50 > 2500 nM T66505 CAI9O3 56675787 IC50 > 2500 nM T66505 CSA35C 56675788 IC50 > 2500 nM T66505 CMKQ61 56675800 IC50 = 1600 nM T66505 CK6GW1 56675801 IC50 = 350 nM T66505 CF2GB3 56675802 IC50 = 3 nM T66505 C6IU9P 56675925 IC50 > 2500 nM T66505 CF3R6A 56675926 IC50 = 1500 nM T66505 C04FDY 56675927 IC50 = 2500 nM T66505 C5I4KA 56676509 IC50 = 21 nM T66505 C6RVC4 56676510 IC50 = 230 nM T66505 C41FSK 56676511 IC50 = 19 nM T66505 CO9AX8 56678641 IC50 = 46 nM T66505 CBZ1S6 56678642 IC50 = 180 nM T66505 CL9V4G 56678643 IC50 = 360 nM T66505 CEI80K 56678644 IC50 = 15 nM T66505 CZ9LW6 56678777 IC50 = 79 nM T66505 CWMH38 56679102 IC50 > 2500 nM T66505 CKN39Z 56679103 IC50 > 2500 nM T66505 C0DV4W 56679122 IC50 = 1800 nM T66505 C07JIH 56679237 IC50 > 2500 nM T66505 CR19BZ 56679238 IC50 = 350 nM T66505 C3MI4V 56679239 IC50 = 1700 nM T66505 CC81YD 56679828 IC50 = 430 nM T66505 C03JCI 56679829 IC50 = 1400 nM T66505 CI6UC5 56680279 IC50 = 7800 nM T66505 CDR92Q 56680280 IC50 = 5100 nM T66505 C06HAF 56681960 IC50 = 370 nM T66505 CS30BK 56681961 IC50 = 16 nM T66505 C1Y0MO 56682216 IC50 = 30 nM T66505 CPRT14 56682402 IC50 = 2100 nM T66505 C07GSV 56682403 IC50 > 2500 nM T66505 CDH41P 56682417 IC50 = 760 nM T66505 CGCH03 56682418 IC50 = 25 nM T66505 C3F6TH 56682550 IC50 = 220 nM T66505 CH46PS 56682551 IC50 = 1400 nM T66505 C7BX5M 56682552 IC50 = 340 nM T66505 CN4RZ3 56682553 IC50 = 280 nM T66505 C3L5PZ 56682554 IC50 > 2500 nM T66505 C14GVW 56683156 IC50 = 140 nM T66505 CV85DJ 56683157 IC50 = 42 nM T66505 C6F7RL 56683158 IC50 = 12 nM T66505 C32GXL 56964691 IC50 = 24 nM T66505 C2Q8VL 56964692 IC50 = 41 nM T66505 C27ION 57326206 IC50 = 100 nM T66505 CRJ90X 57326301 IC50 = 180 nM T66505 CH96BW 57326302 IC50 = 820 nM T66505 CL8H5N 57326385 IC50 = 1100 nM T66505 C7SI0M 57326387 IC50 = 29 nM T66505 C61TYN 57326482 IC50 = 130 nM T66505 CF4X2S 57326483 IC50 = 520 nM T66505 CMI5L4 57326484 IC50 = 1800 nM T66505 C32LFE 67374618 IC50 < 16 nM T66505 C46VLA 67374621 EC50 = 15 nM T66505 CLKN38 67375395 IC50 < 19 nM T66505 C5BFR4 67378301 EC50 = 115 nM T66505 CKB37H 67379186 IC50 < 40 nM T66505 C8M9VH 67379418 EC50 = 28 nM T66505 C07NTU 68747277 IC50 = 42 nM T66505 CD9J0Y 68778068 EC50 = 30 nM T66505 CG16HX 68780878 EC50 = 7 nM T66505 CMGA79 70682196 EC50 = 27 nM T66505 CH0T3O 70684298 EC50 = 89 nM T66505 CTCF71 70688555 EC50 = 22 nM T66505 C1Y7FR 70688556 IC50 > 450 nM T66505 CNER46 70690618 EC50 = 21 nM T66505 CTYA67 70692760 EC50 = 8 nM T66505 CFYG52 70694242 IC50 = 110 nM T66505 C45SUB 70694800 EC50 = 17 nM T66505 C95IBJ 70694801 EC50 = 40 nM T66505 C2SWX1 70696850 EC50 = 29 nM T66505 CO58QT 71458712 Ki = 37.9 nM T66505 C0J3TE 76311001 IC50 = 300 nM T66505 C89CXE 76311004 IC50 = 40 nM T66505 CWZE58 76318208 IC50 = 100 nM T66505 C6H5MS 76848956 Ki = 30 nM T66505 C53NWC 86294818 IC50 = 87 nM T66505 CM0A5R 90286184 IC50 = 1800 nM T66505 CIU6F5 90286320 IC50 = 4100 nM T66505 CJ85YQ 90286388 IC50 > 10000 nM T66505 CW6BO1 90286529 IC50 = 910 nM T66505 C0YEV1 90286574 IC50 = 270 nM T66505 C89TEO 90299606 IC50 = 890 nM T66505 C5V3LH 90299611 IC50 = 350 nM T66505 C7LTZ2 90299612 IC50 = 300 nM T66505 C2UV3X 90299614 IC50 = 440 nM T66505 CZ1GP2 90299621 IC50 = 1300 nM T66505 CKD1F0 90299647 IC50 = 690 nM T66505 CFHB98 90644096 IC50 > 25000 nM T66505 CWK6N7 90656290 IC50 = 2700 nM T66505 CK2I6N 90656291 IC50 = 520 nM T66505 CRI41W 90656292 IC50 = 4100 nM T66505 CL29HQ 90656293 IC50 = 790 nM T66505 CD2PB6 90656294 IC50 > 10000 nM T66505 CS8TB7 90656295 IC50 > 10000 nM T66505 CWL3E0 90656296 IC50 = 550 nM T66505 CW7BV0 90656297 IC50 = 1200 nM T66505 CU4NV3 90656298 IC50 = 1500 nM T66505 CP36FA 90656299 IC50 = 420 nM T66505 C6F9NY 90656300 IC50 = 270 nM T66505 COK94Z 90656301 IC50 = 200 nM T66505 CRG6J5 90656302 IC50 = 380 nM T66505 CR4K2D 90656303 IC50 = 270 nM T66505 C9ZU3G 90656304 IC50 = 740 nM T66505 CI7F1H 90656305 IC50 = 960 nM T66505 CVH8R7 90656306 IC50 = 650 nM T66505 C9WDS7 97046899 Ki = 33 nM T66505 CM7LD8 122185868 IC50 = 5.6 nM T66505 CL0ZB6 122185870 IC50 = 10 nM T66505 C9CZ8G 127039132 IC50 = 19 nM T66505 CDVZ38 127039452 IC50 = 42 nM T66505 CILZ74 127048425 IC50 = 373 nM T66505 C0CF8P 127048730 IC50 = 294 nM T66505 C87LZN 127048731 IC50 = 315 nM T66505 C43IVQ 127048732 IC50 = 18 nM T66505 C38MXE 127048733 IC50 = 192 nM T66505 CS57TL 127048734 IC50 = 135 nM T66505 CDT1A0 127049057 IC50 = 352 nM T66505 C92DBP 127049409 IC50 = 326 nM T66505 C8NO0A 127051279 IC50 = 261 nM T66505 CWT20F 127052154 IC50 = 431 nM T66505 CKM9A3 127052181 IC50 = 217 nM T66505 CP7S9A 127052483 IC50 = 92 nM T66505 CCQ86W 127052484 IC50 = 213 nM T66505 C6LU2S 127052485 IC50 = 56 nM T66505 C2CA0W 127053107 IC50 = 456 nM T66505 C2SAG7 127053109 IC50 = 237 nM T66505 CXI0B3 132578555 IC50 > 10000 nM T66505 CY0BT9 136210502 IC50 = 290 nM T66505 CX67HE 136210503 IC50 = 370 nM T66505 CKP6L1 136210504 IC50 = 70 nM T66505 CL47YD 136210505 IC50 = 220 nM T66505 CE1US4 136210506 IC50 = 70 nM T66505 C7OW0J 136210508 IC50 = 160 nM T66505 CL4IW7 136210509 IC50 = 190 nM T66505 CDFZ95 136210510 IC50 = 33 nM T66505 CKS3V1 136210511 IC50 = 5 nM T66505 CKO48T 136210512 IC50 = 110 nM T66505 CE9OD5 136210517 IC50 = 900 nM T66505 CB7AI4 136210518 IC50 = 14 nM T66505 C0TI5R 136244207 IC50 = 640 nM T66505 C9C5MY 145958866 IC50 = 10 nM T66505 CJ8X4A 155515079 Ki = 55 nM T66505 COKI80 155515124 IC50 = 3.9 nM T66505 CTO9C8 155547338 IC50 = 18 nM T66505 CRG7H3 155549835 Ki = 45 nM T66505 C95DIM 155559226 Ki = 28 nM T66505 D03NPX 447077 Ki = 46.2 nM T66505 D05UKJ 442972 Ki = 12.7 nM T66505 D0R8DO 6404568 IC50 = 4237 nM T66505 D0S5OU 73729049 IC50 = 440 nM T41201 CGNU14 10408898 IC50 = 350 nM T41201 CZIY89 11081290 IC50 = 25 nM T41201 CQ4EM2 44344844 IC50 = 40 nM T41201 CCA3Z7 44344899 IC50 = 20 nM T41201 CTPO43 44345020 IC50 = 6 nM T41201 C5KH6G 44345023 IC50 = 5 nM T41201 CL6KF8 44345101 IC50 = 150 nM T41201 C6T5UV 44345102 IC50 = 45 nM T41201 CL32RO 44345105 IC50 = 10 nM T41201 C18KAP 44345106 IC50 = 100 nM T78319 CKUJ53 16217499 IC50 = 6700000 nM T78319 C5D3HE 30980948 IC50 = 14100000 nM T78319 CH8Z3J 73441667 IC50 = 3500000 nM T78319 CG0O3E 90655419 IC50 = 1320000 nM T78319 CR5MK9 90655420 IC50 = 108000 nM T78319 C3CNA9 90655421 IC50 = 65000 nM T78319 CF0EX8 90655422 IC50 = 48000 nM T78319 CGL84T 90655423 IC50 = 36000 nM T78319 D03EPY 7046 IC50 = 27000000 nM T43721 D02ENG 6918651 IC50 > 10000 nM T43721 D05WCI 11670435 IC50 > 10000 nM T43721 D0B5HF 44476893 IC50 > 10000 nM T43721 D0O1ZI 25006684 IC50 > 30000 nM T43721 D0R8IU 24946280 IC50 > 30000 nM T43721 D0T8QB 14982 IC50 = 0.4 nM T43721 D07EBU 135565424 IC50 > 10000 nM T43721 D07FHW 23725123 IC50 > 500000 nM T43721 CDM6C4 92730 IC50 = 400 nM T43721 C7JEN0 94320 IC50 = 750 nM T43721 C2O8KM 101788 IC50 = 490 nM T43721 CFG6D1 111253 IC50 = 329 nM T43721 C8UQT9 1484979 IC50 > 10000 nM T43721 C34FUY 2953793 Ki > 10000 nM T43721 C3B7LM 3146235 IC50 = 8900 nM T43721 CPT5Y6 6918663 IC50 > 200000 nM T43721 C84RBQ 9797661 IC50 > 4000 nM T43721 CY2K5B 9823394 IC50 = 4000 nM T43721 CHV1E3 9975108 IC50 > 4000 nM T43721 CSL50G 9975639 IC50 > 4000 nM T43721 CDZ92L 9998483 IC50 > 4000 nM T43721 CBUP07 10018475 IC50 = 1270 nM T43721 C0I6WB 10040175 IC50 = 3318 nM T43721 CU1W4M 10040176 IC50 = 2006 nM T43721 C4L0HV 10043410 IC50 > 4000 nM T43721 CA4SJ7 10064183 IC50 > 4000 nM T43721 C5LKO8 10085885 IC50 = 1035 nM T43721 CW6KU4 10250720 IC50 = 1300 nM T43721 CO0H7A 10250842 IC50 > 4000 nM T43721 COT1X3 10308303 IC50 > 4000 nM T43721 C2LWK5 10315044 IC50 > 4000 nM T43721 C0QH6L 10335644 IC50 > 4000 nM T43721 C7IUQ6 10335880 IC50 > 4000 nM T43721 CI64PJ 10340916 IC50 > 4000 nM T43721 CL5X6K 10355633 IC50 > 4000 nM T43721 CTLN27 10357519 IC50 > 4000 nM T43721 CTU13Q 10357992 IC50 = 503 nM T43721 CWKP54 10359991 IC50 > 4000 nM T43721 CEO4C7 10360107 IC50 = 613 nM T43721 CUL28X 10380007 IC50 < 4000 nM T43721 CF4NL2 10381554 IC50 = 216 nM T43721 CR4V3G 10402262 IC50 > 4000 nM T43721 C65EQT 10403095 IC50 = 1037 nM T43721 CV8K3E 10446474 IC50 = 4000 nM T43721 CQ9X4Y 10446475 IC50 > 4000 nM T43721 CYI70T 10447474 IC50 = 4000 nM T43721 CS06QG 10452320 IC50 > 100000 nM T43721 CA89WN 10470037 IC50 > 4000 nM T43721 C6LJI0 10473292 IC50 > 4000 nM T43721 CXH39G 10474399 IC50 > 4000 nM T43721 C0C6KD 11190936 IC50 = 122 nM T43721 CD3H7R 11232699 IC50 > 200000 nM T43721 C1PKI0 11257147 IC50 > 200000 nM T43721 CW1T5X 11259177 IC50 = 228 nM T43721 CH12WK 11278558 IC50 > 4000 nM T43721 CP9O5R 11280328 IC50 > 200000 nM T43721 CH85OD 11319723 IC50 = 2350 nM T43721 C8FQ9B 11375180 IC50 = 3950 nM T43721 CS0P1Q 11478969 IC50 = 280 nM T43721 CR4I9H 11484764 IC50 = 290 nM T43721 CN08AP 11495851 IC50 > 10000 nM T43721 CLT1Z9 11502804 IC50 = 6300 nM T43721 C76STL 11504178 IC50 = 21000 nM T43721 C19BYP 11505338 IC50 = 50000 nM T43721 CHW7L1 11510573 IC50 > 100000 nM T43721 CE40MU 11524868 IC50 = 550 nM T43721 C8NP4Y 11526147 IC50 = 3 nM T43721 CG1HB5 11533520 IC50 = 24000 nM T43721 CZE42S 11540388 IC50 = 13000 nM T43721 CN1A6F 11540493 IC50 > 100000 nM T43721 C3LVE2 11545617 IC50 = 30000 nM T43721 CD17CO 11551576 IC50 > 10000 nM T43721 CP8L9K 11552169 IC50 = 23000 nM T43721 CCT0Q7 11552781 IC50 = 18000 nM T43721 CA25ZF 11555218 IC50 = 34000 nM T43721 CJ58XB 11576524 IC50 = 25000 nM T43721 CKF3J6 11604308 IC50 = 16000 nM T43721 CGD7X9 11610822 IC50 = 12000 nM T43721 CDL39R 11613794 IC50 > 30000 nM T43721 C7KBZ4 11618761 IC50 = 5500 nM T43721 CW2XN3 11626362 IC50 = 85000 nM T43721 CXS05L 11627334 IC50 > 10000 nM T43721 CMF3U5 11634114 IC50 > 100000 nM T43721 CDL94B 11649095 IC50 > 100000 nM T43721 CX17LY 11654021 IC50 = 1800 nM T43721 C3B4SN 11655097 IC50 > 20000 nM T43721 C1DJ7W 11655188 IC50 = 26000 nM T43721 C1T6KE 11666874 IC50 = 8300 nM T43721 CFH6G5 11670914 IC50 = 20000 nM T43721 CU5TI1 11676805 IC50 > 100000 nM T43721 CJ13XD 11698697 IC50 = 5300 nM T43721 C26ITU 11699075 IC50 = 27000 nM T43721 CK8BF3 11705872 IC50 > 10000 nM T43721 C4D6YM 11712182 IC50 = 60000 nM T43721 C5AT6X 11722880 IC50 = 1961 nM T43721 CO32UM 11724534 IC50 = 1964 nM T43721 C6TPR1 11739354 IC50 > 4000 nM T43721 C4B5XT 11741200 IC50 > 4000 nM T43721 CB9WI2 11742158 IC50 > 4000 nM T43721 C37IRX 11771845 IC50 = 183 nM T43721 C2XW0P 11853305 IC50 = 6040 nM T43721 C4FKP2 13994830 IC50 > 1000000 nM T43721 CEYW48 15953464 IC50 = 2520 nM T43721 CY3A6Q 15987396 IC50 > 10000 nM T43721 C29ACV 15987476 IC50 > 10000 nM T43721 CS1XM4 16049788 IC50 = 100000 nM T43721 C2T4IM 16222378 IC50 = 30.4 nM T43721 C13TPH 16721119 IC50 > 10000 nM T43721 C2OJC1 16726072 IC50 > 10000 nM T43721 C69QUM 20724870 IC50 = 1174 nM T43721 C51LGI 20724898 IC50 > 4000 nM T43721 CP7JM8 20724899 IC50 > 4000 nM T43721 C31VAH 20724901 IC50 > 4000 nM T43721 CJU3T5 20724903 IC50 > 4000 nM T43721 CLX5A8 20724912 IC50 > 4000 nM T43721 CQ6CF3 20755069 IC50 > 4000 nM T43721 CTRD81 20755103 IC50 > 1000 nM T43721 CD1SR0 22591684 IC50 > 4000 nM T43721 CQ6AO5 22591709 IC50 = 7.5 nM T43721 CWF51V 22591726 IC50 > 4000 nM T43721 CEB47A 24744047 IC50 = 21200 nM T43721 CGR84K 24854349 IC50 > 500000 nM T43721 C6BV8N 24854350 IC50 > 500000 nM T43721 CEW31B 24856362 IC50 > 100000 nM T43721 C7QU2Z 24883422 IC50 = 10000 nM T43721 CLYS75 24889741 IC50 = 20 nM T43721 CVD4K7 24889906 IC50 = 15000 nM T43721 C6EFK9 24889907 IC50 > 30000 nM T43721 C5QD7L 24890069 IC50 = 1600 nM T43721 C9XUC0 24890070 IC50 = 1800 nM T43721 C3A9HI 24890073 IC50 = 90000 nM T43721 C6IHL0 24890239 IC50 = 23000 nM T43721 CEV27L 24895554 IC50 > 10000 nM T43721 C8LYV0 24895658 IC50 > 10000 nM T43721 C2QWU0 24895661 IC50 > 10000 nM T43721 C1G6DM 24895969 IC50 > 10 nM T43721 C59MRG 24896012 IC50 > 10 nM T43721 C6UYQ4 24948172 IC50 > 10000 nM T43721 CJL38O 25065024 IC50 > 10000 nM T43721 C8GR2K 25065025 IC50 = 510 nM T43721 CEMG39 25065027 IC50 > 10000 nM T43721 CB36SV 25065227 IC50 > 10000 nM T43721 C7YH6J 25065230 IC50 > 10000 nM T43721 C9EQ1D 25065231 IC50 > 10000 nM T43721 CU12CJ 25065232 IC50 = 10 nM T43721 CEQF65 25210659 IC50 > 100000 nM T43721 CU7E9B 25265683 IC50 > 10000 nM T43721 CMVE89 42603038 IC50 > 10000 nM T43721 C6VQM9 44143289 IC50 > 100000 nM T43721 CZ58CY 44143291 IC50 > 100000 nM T43721 C8X2ZV 44143292 IC50 > 100000 nM T43721 C1IA7U 44143299 IC50 > 100000 nM T43721 C63STN 44196869 IC50 = 31.2 nM T43721 C7YTM0 44197230 IC50 > 4000 nM T43721 CHA7J4 44250316 IC50 > 1000000 nM T43721 C9S2HX 44402393 IC50 > 200000 nM T43721 C8C2QJ 44402534 IC50 > 200000 nM T43721 CW7IP2 44402550 IC50 > 200000 nM T43721 C0NUI2 44402662 IC50 > 200000 nM T43721 C42FXZ 44418375 IC50 > 100000 nM T43721 CC93VQ 44418376 IC50 = 16000 nM T43721 CP9DO4 44418378 IC50 = 52000 nM T43721 CR7K6S 44418382 IC50 > 100000 nM T43721 C7B6GT 44418383 IC50 > 100000 nM T43721 C1Q8CH 44418384 IC50 > 100000 nM T43721 C7JNH9 44418385 IC50 = 100000 nM T43721 CB58SX 44418389 IC50 = 70000 nM T43721 CGKR51 44418390 IC50 = 49000 nM T43721 CQT37N 44418391 IC50 > 100000 nM T43721 CED27U 44418395 IC50 > 100000 nM T43721 C9L7BU 44418396 IC50 > 100000 nM T43721 C28DBM 44418400 IC50 > 100000 nM T43721 C1KD8E 44418401 IC50 > 100000 nM T43721 CT79UX 44418408 IC50 > 100000 nM T43721 C7RW1O 44418409 IC50 > 100000 nM T43721 C7WQD4 44418433 IC50 > 30000 nM T43721 CV87RE 44418434 IC50 > 30000 nM T43721 CK74ZJ 44418441 IC50 > 30000 nM T43721 C02AMZ 44418445 IC50 > 30000 nM T43721 C7YCN4 44418447 IC50 > 100000 nM T43721 C7AKJ2 44418450 IC50 > 100000 nM T43721 C90QWN 44418451 IC50 = 55000 nM T43721 CA2J1I 44418452 IC50 = 11000 nM T43721 CE1W9Y 44418456 IC50 = 90000 nM T43721 C7R3AT 44418457 IC50 > 100000 nM T43721 C4MVN6 44418458 IC50 = 15000 nM T43721 CXFR60 44418459 IC50 = 100000 nM T43721 CAW7Z2 44418817 IC50 > 100000 nM T43721 CC8ZR0 44418821 IC50 > 100000 nM T43721 CKX95Y 44418852 IC50 > 100000 nM T43721 CF56NG 44418856 IC50 = 56000 nM T43721 CGX84K 44418857 IC50 = 62000 nM T43721 CSP8W1 44419286 IC50 > 30000 nM T43721 CQH6X0 44419304 IC50 = 17000 nM T43721 CBI64W 44419309 IC50 = 14000 nM T43721 C6LOU9 44419313 IC50 = 630 nM T43721 C32WUT 44420153 IC50 > 10000 nM T43721 C14JQE 44420164 IC50 > 10000 nM T43721 C76RGZ 44420166 IC50 > 10000 nM T43721 CINJ57 44420180 IC50 > 10000 nM T43721 CWM5F9 44420181 IC50 > 10000 nM T43721 CLA82E 44420186 IC50 > 10000 nM T43721 C0ET3O 44420190 IC50 > 10000 nM T43721 C3JF5Z 44420196 IC50 > 10000 nM T43721 C64UQO 44420202 IC50 > 10000 nM T43721 CJI76N 44420207 IC50 > 10000 nM T43721 C0T6ML 44420212 IC50 > 10000 nM T43721 C5Y4UB 44420215 IC50 > 10000 nM T43721 C1NCR3 44420232 IC50 > 10000 nM T43721 CQ7B8C 44420233 IC50 > 10000 nM T43721 C0X3PE 44420237 IC50 > 10000 nM T43721 CO4S5M 44420238 IC50 > 10000 nM T43721 CV6P7Y 44420242 IC50 > 10000 nM T43721 C8IH5C 44420243 IC50 > 10000 nM T43721 CZG60J 44420244 IC50 = 50000 nM T43721 CN2B1J 44420246 IC50 > 10000 nM T43721 CG90VX 44420247 IC50 > 10000 nM T43721 C5PU7K 44420248 IC50 > 10000 nM T43721 C7KW0L 44420249 IC50 = 100000 nM T43721 CBL6K2 44420251 IC50 > 10000 nM T43721 CF9N4T 44420252 IC50 > 10000 nM T43721 CVX2Z3 44420253 IC50 > 10000 nM T43721 CX8IQ0 44420257 IC50 > 10000 nM T43721 CN3W4S 44420259 IC50 = 3600 nM T43721 C1YLR4 44420285 IC50 = 65000 nM T43721 CNRY91 44420288 IC50 > 10000 nM T43721 CF23SE 44420291 IC50 > 10000 nM T43721 CE7T4W 44420294 IC50 = 15000 nM T43721 CJ1O7N 44438556 IC50 = 17000 nM T43721 CH0K4M 44438559 IC50 = 3500 nM T43721 CXM65L 44438562 IC50 = 26000 nM T43721 CM01KY 44438566 IC50 = 20000 nM T43721 CFLP12 44438567 IC50 = 12000 nM T43721 CAW10E 44438568 IC50 = 25000 nM T43721 C3IK2C 44438569 IC50 > 100000 nM T43721 C43RLG 44438570 IC50 = 580 nM T43721 CM1Y7N 44438669 IC50 = 15000 nM T43721 CUE3I1 44438670 IC50 = 3300 nM T43721 CQM10L 44438671 IC50 = 15000 nM T43721 CB19EU 44438672 IC50 = 5400 nM T43721 CL4Y3J 44438673 IC50 = 17000 nM T43721 C7ON6I 44438675 IC50 = 65000 nM T43721 C5LN8W 44438676 IC50 > 100000 nM T43721 C8VI7M 44438677 IC50 > 100000 nM T43721 CV12KJ 44438678 IC50 = 21000 nM T43721 CBX9L4 44438679 IC50 = 59000 nM T43721 CF5YU4 44438681 IC50 > 100000 nM T43721 CJ2M3L 44438682 IC50 = 9000 nM T43721 CJB5H3 44443435 Ki > 10000 nM T43721 C3U1WZ 44448872 IC50 > 4000 nM T43721 CZ5A6G 44576636 IC50 > 4000 nM T43721 CHD6G5 44576637 IC50 > 4000 nM T43721 CK67LT 44576651 IC50 > 4000 nM T43721 C9JB2Y 44576672 IC50 > 4000 nM T43721 CMJ91U 44576707 IC50 > 4000 nM T43721 C8D1LU 44576749 IC50 > 4000 nM T43721 CKH1A8 44576750 IC50 > 4000 nM T43721 CN93WV 44576751 IC50 > 4000 nM T43721 CAH82I 44576752 IC50 > 4000 nM T43721 CK5S4W 44576802 IC50 > 4000 nM T43721 C9L3CP 44576803 IC50 > 4000 nM T43721 C2F5RM 44576804 IC50 > 4000 nM T43721 CK41XQ 44576805 IC50 > 4000 nM T43721 CO5YU9 44576846 IC50 > 4000 nM T43721 C4YIR7 44576873 IC50 > 4000 nM T43721 C2HW0I 44576875 IC50 > 4000 nM T43721 COQ7U4 44576945 IC50 > 4000 nM T43721 C18JAM 45269430 IC50 > 1000000 nM T43721 CGPF36 45270351 IC50 > 10000 nM T43721 C83OJH 45271081 IC50 > 1000000 nM T43721 C7O3DH 45271171 IC50 = 2487 nM T43721 CE07FS 45272366 IC50 > 10000 nM T43721 CK65BP 46213656 IC50 > 10000 nM T43721 CHI5S0 46216688 IC50 > 10000 nM T43721 CAX31B 46216689 IC50 > 10000 nM T43721 CN39HK 46229717 IC50 = 268 nM T43721 C4N8DB 46231719 IC50 > 10000 nM T43721 C4WT0Q 46231721 IC50 = 9000 nM T43721 CIX36V 46894126 IC50 = 2.9 nM T43721 CS13YQ 49846481 IC50 > 100000 nM T43721 C6W2XQ 49846838 IC50 > 100000 nM T43721 CA8N9P 52911994 IC50 > 30000 nM T43721 CICZ45 52918012 IC50 > 10000 nM T43721 C4X2WF 52939227 IC50 = 11 nM T43721 CQ6R0S 52939228 IC50 = 33 nM T43721 C1YRT3 52940913 IC50 = 4.9 nM T43721 CSXY62 52941059 IC50 = 7350 nM T43721 C8X4NE 52945350 IC50 = 61.1 nM T43721 CE3AQ9 52945888 IC50 = 458 nM T43721 CO7ZR1 52947102 IC50 = 8650 nM T43721 C2KHL7 52947144 IC50 = 14.5 nM T43721 CJI28A 52950107 IC50 = 2130 nM T43721 CSUK37 53322740 IC50 = 104 nM T43721 CQ7J8E 53322756 IC50 = 194 nM T43721 C6W3JM 53326660 IC50 = 17 nM T43721 CP91BU 53326661 IC50 = 45 nM T43721 C9H5YE 53361128 IC50 > 10000 nM T43721 CN93FS 54580118 IC50 > 4000 nM T43721 CF05VK 54580143 IC50 > 4000 nM T43721 C7FXV6 54580144 IC50 > 4000 nM T43721 C2M8XQ 54580210 IC50 > 4000 nM T43721 C4Q6MO 54580243 IC50 > 4000 nM T43721 CBX17R 54581094 IC50 > 4000 nM T43721 C8O9WK 54581095 IC50 > 4000 nM T43721 CM67RK 54581096 IC50 = 2300 nM T43721 C8ZDF3 54581137 IC50 > 4000 nM T43721 C14YRS 54581213 IC50 > 4000 nM T43721 CQ7GV2 54582134 IC50 > 4000 nM T43721 CZ1B6L 54582135 IC50 > 4000 nM T43721 C07KDH 54582136 IC50 = 3100 nM T43721 CK29GC 54582137 IC50 > 4000 nM T43721 CKGX19 54582164 IC50 > 4000 nM T43721 CWA6Q0 54582242 IC50 > 4000 nM T43721 C07LYE 54582261 IC50 > 4000 nM T43721 CP2N1C 54582262 IC50 > 4000 nM T43721 CM2QX4 54583079 IC50 > 4000 nM T43721 CMKQ26 54583080 IC50 > 4000 nM T43721 C2G7LK 54583125 IC50 > 4000 nM T43721 CL6Z9X 54583126 IC50 > 4000 nM T43721 CGM2W4 54583127 IC50 > 4000 nM T43721 CF42QY 54583128 IC50 > 4000 nM T43721 CWHS39 54583210 IC50 = 4000 nM T43721 CDK5V0 54583231 IC50 > 4000 nM T43721 C5V4DY 54583232 IC50 > 4000 nM T43721 C1JV9N 54583233 IC50 = 1600 nM T43721 CKA9L3 54583234 IC50 > 4000 nM T43721 CZ4YV3 54584081 IC50 > 4000 nM T43721 CHP62C 54584119 IC50 > 4000 nM T43721 CD2QO1 54584120 IC50 = 1300 nM T43721 CCT0B2 54584121 IC50 > 4000 nM T43721 C0VPS6 54584122 IC50 > 4000 nM T43721 C6P5XR 54584196 IC50 > 4000 nM T43721 CY2WM3 54584197 IC50 > 4000 nM T43721 CXNP26 54584198 IC50 > 4000 nM T43721 CWY83C 54584415 IC50 > 4000 nM T43721 CGD4N3 54585028 IC50 > 4000 nM T43721 C8NZ2B 54585029 IC50 > 4000 nM T43721 CHW48S 54585030 IC50 > 4000 nM T43721 CZ8R0S 54585053 IC50 > 4000 nM T43721 C04IZR 54585054 IC50 > 4000 nM T43721 C6GZB9 54585157 IC50 > 4000 nM T43721 C5SHO2 54585992 IC50 > 4000 nM T43721 CJA5Z6 54585993 IC50 > 4000 nM T43721 C4JTZ5 54585994 IC50 > 4000 nM T43721 CKF15E 54586030 IC50 > 4000 nM T43721 CT12RX 54586031 IC50 > 4000 nM T43721 CD6FC5 54586091 IC50 = 1300 nM T43721 CDG95F 54586092 IC50 > 4000 nM T43721 CJ8K1Y 54586966 IC50 > 4000 nM T43721 C51MDN 54586967 IC50 > 4000 nM T43721 CH2F8P 54586968 IC50 > 4000 nM T43721 C61ZTA 54586969 IC50 > 4000 nM T43721 C3Y6HF 54587012 IC50 > 4000 nM T43721 CUF68X 54587090 IC50 = 460 nM T43721 CI1PV5 54587121 IC50 > 4000 nM T43721 C6PSJ3 54587122 IC50 > 4000 nM T43721 C9D1UH 54587123 IC50 > 4000 nM T43721 C82TDJ 54587124 IC50 > 4000 nM T43721 CNQ41E 54590876 IC50 > 10000 nM T43721 C3IAB0 57392785 IC50 = 386 nM T43721 C4I9DE 57408764 IC50 > 100000 nM T43721 CM2DN9 57408765 IC50 = 400 nM T43721 CAI0P1 57418438 IC50 > 100000 nM T43721 C39SNL 57916360 IC50 > 30000 nM T43721 CG16CV 57916503 IC50 > 30000 nM T43721 CG1Y8Z 67464068 IC50 > 10000 nM T43721 CJL0P9 67468231 IC50 > 10000 nM T43721 CM80QX 70687773 EC50 = 2200 nM T43721 CZI43B 70691963 EC50 = 860 nM T43721 CQ5GB9 70691964 EC50 = 720 nM T43721 C3CAB4 71456572 IC50 = 2200 nM T43721 CU24OM 71458421 IC50 > 10000 nM T43721 C0D3IO 71511561 IC50 > 10 nM T43721 C4LAB0 72204152 IC50 = 2200 nM T43721 C17NBW 72204153 IC50 = 2410 nM T43721 CTN6U7 72204155 IC50 = 2690 nM T43721 C0N7EJ 72204340 IC50 = 5850 nM T43721 CS3TL6 72204534 IC50 = 4210 nM T43721 CA5KC4 72204732 IC50 = 6760 nM T43721 C2Q6YJ 72670421 IC50 = 4000 nM T43721 CYAJ36 73345978 IC50 = 1600 nM T43721 CG15WM 73352110 IC50 > 100000 nM T43721 CALM65 73352112 IC50 > 100000 nM T43721 C9WA7F 73353568 IC50 > 100000 nM T43721 CV72YC 73355069 IC50 > 100000 nM T43721 CGR3P5 73355072 IC50 = 228700 nM T43721 C15SEC 73356624 IC50 > 1000000 nM T43721 C2FOM5 73356626 IC50 = 700 nM T43721 CV70BR 73356628 IC50 > 1000000 nM T43721 CWC4Z5 73356629 IC50 > 100000 nM T43721 CPN65E 90643787 IC50 > 30000 nM T43721 CQ23WR 90667215 IC50 > 30000 nM T43721 CFSK10 101911911 IC50 = 25500 nM T43721 CO0H9S 101911912 IC50 = 40700 nM T43721 C91CLR 101911913 IC50 = 299600 nM T43721 C9RBA1 101911914 IC50 = 283600 nM T43721 CMOG09 101911915 IC50 = 11300 nM T43721 CMX6S5 118709259 IC50 > 10000 nM T43721 C7WYI8 127037831 IC50 > 1000000 nM T43721 CI5HA6 127037875 IC50 > 1000000 nM T43721 CP0JV9 127038197 IC50 > 1000000 nM T43721 C4E1LF 127040565 IC50 > 1000000 nM T43721 CTN4E7 127040566 IC50 > 1000000 nM T43721 CB67LT 127040901 IC50 > 1000000 nM T43721 C5P3KE 127040902 IC50 > 1000000 nM T43721 CT5Q1A 127040903 IC50 > 1000000 nM T43721 CW3FN4 127040904 IC50 > 1000000 nM T43721 C9EQX2 127040905 IC50 > 1000000 nM T43721 C32ADQ 127040906 IC50 > 1000000 nM T43721 CYNI06 127041808 IC50 > 1000000 nM T43721 C1ZUD5 127041809 IC50 > 1000000 nM T43721 CCU4H6 127041810 IC50 > 1000000 nM T43721 CZN2A0 127041811 IC50 > 1000000 nM T43721 CCKL17 127042099 IC50 > 1000000 nM T43721 C24EQS 127042100 IC50 > 1000000 nM T43721 CE64CI 127042101 IC50 > 1000000 nM T43721 COR6A5 127042102 IC50 > 1000000 nM T43721 CKM3I9 127042477 IC50 > 1000000 nM T43721 CMP75K 127042478 IC50 > 1000000 nM T43721 CMCP64 127042780 IC50 > 1000000 nM T43721 C4OUL9 127042781 IC50 > 1000000 nM T43721 CGWV92 132053849 IC50 < 100 nM T43721 CT05EL 135399889 IC50 > 10000 nM T43721 C02KAD 135440148 IC50 > 4000 nM T43721 CE0S3Y 135465949 IC50 > 4000 nM T43721 CM7A1J 135492551 IC50 > 4000 nM T43721 C98OIC 135611051 IC50 > 10000 nM T43721 CCQJ43 135611106 IC50 > 10000 nM T43721 C2K9OD 135611129 IC50 > 10000 nM T43721 C4YO9E 135612240 IC50 > 4000 nM T43721 C76MEG 135783319 IC50 > 10000 nM T43721 CMQ2L1 135783320 IC50 > 10000 nM T43721 CE6L4S 135783321 IC50 > 10000 nM T43721 CTAM34 135783322 IC50 > 10000 nM T43721 C7B3JV 135783325 IC50 > 10000 nM T43721 C59KXI 135783328 IC50 > 10000 nM T43721 CKB54L 135783329 IC50 > 10000 nM T43721 C7ZTC5 135783333 IC50 > 10000 nM T43721 C09UQY 135783334 IC50 > 10000 nM T43721 CL5F0J 135783335 IC50 > 10000 nM T43721 CA2ZD0 135857035 IC50 > 10000 nM T43721 CV64MY 135857036 IC50 > 10000 nM T43721 C6IYH3 135967877 IC50 = 35000 nM T43721 C0FO4G 135980568 IC50 = 15 nM T43721 CX3VU1 136000590 IC50 > 4000 nM T43721 CNQ25Z 136021384 IC50 > 10000 nM T43721 C7W4GE 136088954 IC50 > 4000 nM T43721 CT3RN8 136141565 IC50 = 11 nM T43721 CR74OZ 136188845 IC50 > 4000 nM T43721 CWJ0X4 137637923 IC50 = 6261 nM T43721 CDS86M 137656441 IC50 = 9582 nM T43721 C94RSY 137656587 IC50 > 10000 nM T43721 C0DHM9 145952000 IC50 = 100 nM T43721 CC91LF 145952333 IC50 < 100 nM T43721 CDT3Q6 145956314 IC50 = 1000 nM T43721 C09QUS 145958039 IC50 < 100 nM T43721 CV6Q5J 145960157 IC50 = 100 nM T43721 CMVS94 155512106 IC50 > 500000 nM T43721 C1F9PV 155515115 IC50 > 500000 nM T43721 CPO9M4 155520336 IC50 > 500000 nM T43721 CXOU89 155521135 IC50 > 500000 nM T43721 C8WNT0 155521284 IC50 > 500000 nM T43721 CN59WH 155525513 IC50 > 500000 nM T43721 C1D4WM 155537728 IC50 > 500000 nM T43721 CV5KQ0 155543491 IC50 > 500000 nM T43721 CKFU03 155545095 IC50 > 500000 nM T43721 CG19XT 155548236 IC50 > 500000 nM T43721 CB08IM 155548826 IC50 > 500000 nM T43721 C1GC0O 155553184 IC50 > 500000 nM T43721 CEM03Y 155556588 IC50 > 500000 nM T43721 C9E6AM 155561480 IC50 > 500000 nM T43721 COWH25 155562798 IC50 > 500000 nM T43721 CZT7P4 155567250 IC50 > 500000 nM T43721 D00PSW 3630776 IC50 > 3000 nM T43721 D00QOL 11673314 IC50 > 10000 nM T43721 D02KXX 586971 IC50 > 200000 nM T43721 D02WUU 15627039 IC50 > 200000 nM T43721 D03JWH 135450677 IC50 > 10000 nM T43721 D04WVV 10193044 IC50 > 4000 nM T43721 D0A4ZR 135950111 Ki > 10000 nM T43721 D0EU9W 16750524 IC50 > 200000 nM T43721 D0L4VR 636403 IC50 = 170 nM T43721 D0M4PP 4271571 IC50 > 200000 nM T43721 D0P7RN 1483401 IC50 > 200000 nM T43721 D0T3FW 44419251 IC50 > 10000 nM T43721 D0U8IF 10114 IC50 = 1.2 nM T09513 D0A3MV 448014 IC50 > 100000 nM T09513 CH20NR 403176 IC50 = 20 nM T09513 CNG96H 25210579 IC50 > 10000 nM T09513 CE1ZK6 54759168 IC50 > 10000 nM T09513 CL5IR0 135512024 IC50 = 7 nM T09513 D03YVL 5472558 IC50 = 25000 nM T09513 D0Y0ES 3707 IC50 = 100 nM T32880 D06VNK 1110 IC50 = 3000 nM T32880 D01SPD 69669724 IC50 = 280 nM T32880 D03GOO 444972 IC50 = 19000 nM T32880 D03YKE 11256664 IC50 = 591.4 nM T32880 D07KEH 23634441 IC50 = 29 nM T32880 D0N6CS 6914666 IC50 = 70 nM T32880 D00IKR 52912218 IC50 = 14000 nM T32880 D01XZT 24891734 IC50 = 650 nM T32880 D03TPE 97394 IC50 = 14000 nM T32880 D09NCT 53392492 IC50 = 83000 nM T32880 D0QI0J 134204791 IC50 = 15000 nM T32880 CWJ0U1 5312 IC50 = 18000 nM T32880 CMO39B 7493 Ki > 300000 nM T32880 CK23OU 76549 IC50 > 1000000 nM T32880 C8JBE5 94284 IC50 = 8500 nM T32880 C06WZQ 222878 IC50 > 100000 nM T32880 CBZ21G 231363 IC50 > 100000 nM T32880 COS62U 245007 IC50 > 100000 nM T32880 C0MHV8 252439 IC50 = 94000 nM T32880 C3OZ5L 919929 IC50 > 100000 nM T32880 C2OS3W 2238068 IC50 > 100000 nM T32880 CHV8N5 4666803 IC50 > 40000 nM T32880 CGP0X9 6914624 IC50 = 1400 nM T32880 CS7C1Z 8027170 IC50 = 12000 nM T32880 CYJ23Z 10470802 IC50 = 4800 nM T32880 CP76HX 11372202 IC50 = 2400 nM T32880 CM6Q3H 11788622 IC50 > 100000 nM T32880 CDM30S 13770962 IC50 > 1000000 nM T32880 CO03CL 14991438 IC50 = 95000 nM T32880 C9M2AL 16126655 IC50 = 190 nM T32880 CIU0N5 16126706 IC50 = 3900 nM T32880 CI45OC 16126774 IC50 = 3600 nM T32880 CX5VP0 18372521 IC50 = 5300 nM T32880 C52JUB 18372631 IC50 = 4400 nM T32880 CN2HO1 18632368 IC50 = 69700 nM T32880 CDSM62 20816892 IC50 = 4200 nM T32880 C20YQO 22122176 IC50 > 1000000 nM T32880 C92REF 22345738 IC50 = 398000 nM T32880 CCAM68 22959876 IC50 > 100000 nM T32880 CGE7Y9 23260762 IC50 > 1000000 nM T32880 CZ9X6U 24812792 IC50 = 3 nM T32880 CZ8WG7 24831508 IC50 = 22.2 nM T32880 CE9N0S 24891150 IC50 > 100000 nM T32880 CV17FS 24894050 IC50 = 21 nM T32880 C0R7YW 25105470 IC50 = 3 nM T32880 C9TN1M 25105471 IC50 = 3 nM T32880 C9CLE1 25138008 IC50 > 1000000 nM T32880 C8P4AV 25173259 IC50 = 185 nM T32880 C5PJZ9 25173339 IC50 = 44 nM T32880 CIM16Z 25173590 IC50 = 7.8 nM T32880 CP8D4L 25173666 IC50 = 140 nM T32880 CTNC06 25173744 IC50 = 52 nM T32880 C92CGK 25173747 IC50 = 30 nM T32880 C5YWM9 25173822 IC50 = 17 nM T32880 CIF90R 25173824 IC50 = 4.1 nM T32880 C3C0AO 25173900 IC50 = 11 nM T32880 C4TNI3 25206050 IC50 = 1500 nM T32880 CS6N9A 42639237 IC50 = 45500 nM T32880 C2AG1B 42639238 IC50 = 8600 nM T32880 C4LK0F 42639413 IC50 = 700 nM T32880 CY6M3D 42639898 IC50 = 1900 nM T32880 CDE5U3 44419123 IC50 = 46000 nM T32880 CFI5L3 44419124 IC50 = 39000 nM T32880 C0U8JS 44419131 IC50 = 15000 nM T32880 C0Y2EG 44419132 IC50 > 100000 nM T32880 CMD26E 44419133 IC50 = 20000 nM T32880 CLQ71X 44419139 IC50 = 4900 nM T32880 C7MYD0 44419140 IC50 = 6500 nM T32880 C0O3EP 44419147 IC50 = 15000 nM T32880 C5IQT0 44419154 IC50 = 18000 nM T32880 CO8HT3 44419159 IC50 = 15000 nM T32880 CGW2A6 44419160 IC50 = 7300 nM T32880 C6ZYP0 44419165 IC50 = 6800 nM T32880 CB1YA2 44419171 IC50 = 19000 nM T32880 C4QH8U 44419179 IC50 = 10000 nM T32880 CY4NW1 44419252 IC50 = 17000 nM T32880 C6T3AY 44419262 IC50 = 5000 nM T32880 C2FSX3 44419264 IC50 = 14200 nM T32880 C5M4KV 44419265 IC50 = 6800 nM T32880 CE5N3Y 44419266 IC50 = 4600 nM T32880 CQ0IJ2 44419267 IC50 = 7400 nM T32880 C38SEB 44419270 IC50 = 16000 nM T32880 C6OR8X 44419271 IC50 = 4400 nM T32880 C0CW1M 44419272 IC50 = 28700 nM T32880 CQ0A4B 44419273 IC50 = 6000 nM T32880 CVE69C 44419277 IC50 = 9700 nM T32880 C7UOR2 44419278 IC50 = 6100 nM T32880 C1H6FT 44419280 IC50 = 8100 nM T32880 CX43WB 44419281 IC50 = 5900 nM T32880 C0YGE2 44419282 IC50 = 14000 nM T32880 CNR45T 44419283 IC50 = 4100 nM T32880 CE5N6U 44419284 IC50 = 10000 nM T32880 C4UEG7 44419285 IC50 = 3200 nM T32880 CGSN20 44419287 IC50 = 7200 nM T32880 COR69J 44419288 IC50 = 6900 nM T32880 C6NXA4 44419290 IC50 = 5800 nM T32880 C3IW5O 44419297 IC50 = 19000 nM T32880 CAP3T5 44419302 IC50 = 24000 nM T32880 C2X1ZV 44419317 IC50 = 2700 nM T32880 CNV8A6 44419318 IC50 = 580 nM T32880 CS85EJ 44419319 IC50 = 1700 nM T32880 CI2M5C 44419320 IC50 = 2400 nM T32880 C0TIU7 44419321 IC50 = 2400 nM T32880 C1MOH2 44419325 IC50 = 1600 nM T32880 C7KUX4 44419326 IC50 = 1600 nM T32880 C37UJB 44419329 IC50 = 2100 nM T32880 C8SQT3 44419330 IC50 = 2900 nM T32880 C2GTJ8 44419333 IC50 = 1700 nM T32880 C96OKR 44419334 IC50 = 2800 nM T32880 CP42UL 44419336 IC50 = 12000 nM T32880 CPX3V9 44419342 IC50 = 24000 nM T32880 C0B9TD 44419346 IC50 > 100000 nM T32880 C5Z3XD 44462724 IC50 = 1.6 nM T32880 C3CST2 44462748 IC50 = 6.8 nM T32880 CR05QL 44469096 IC50 > 100000 nM T32880 C9MK8J 44469097 IC50 = 12589.25 nM T32880 CK6O8G 44469099 IC50 = 19952.62 nM T32880 CADR40 44469101 IC50 = 25118.86 nM T32880 CBSI48 44469229 IC50 = 50118.72 nM T32880 C4U5RZ 44478798 IC50 = 79.43 nM T32880 CR21XB 44478800 IC50 = 158.49 nM T32880 CXOU61 44481885 IC50 = 1000 nM T32880 CCGJ52 44482164 IC50 = 79.43 nM T32880 CIK17O 44482165 IC50 = 398.11 nM T32880 CBL07Q 44482167 IC50 = 398.11 nM T32880 C42FTP 44482169 IC50 = 316.23 nM T32880 CT15UI 44514766 IC50 = 2.1 nM T32880 CW9OQ6 44568201 IC50 = 72 nM T32880 CF9QX3 44568202 IC50 > 40000 nM T32880 CEQL05 44568203 IC50 > 40000 nM T32880 CVWD50 44568204 IC50 = 1300 nM T32880 CX8B7T 44568205 IC50 = 72 nM T32880 CJ12AH 44568206 IC50 = 98 nM T32880 CC4B5M 44568207 IC50 = 33 nM T32880 CU63MS 44568208 IC50 = 27 nM T32880 C69PMH 44568247 IC50 > 40000 nM T32880 C1M3GY 44568248 IC50 = 400 nM T32880 C3JLM8 44568249 IC50 = 410 nM T32880 CF1E4K 44568250 IC50 = 2300 nM T32880 CX2YE1 44568251 IC50 = 21 nM T32880 CO50XS 44568252 IC50 = 11 nM T32880 C43BDN 44568281 IC50 = 4400 nM T32880 CXR89P 44568282 IC50 = 1700 nM T32880 CVID82 44568283 IC50 > 40000 nM T32880 C9JGC4 44568284 IC50 = 600 nM T32880 CG62EN 44568285 IC50 = 50 nM T32880 CK3SI1 44579681 IC50 = 570 nM T32880 CDAN35 44579682 IC50 = 290 nM T32880 CL9O6W 44579683 IC50 = 320 nM T32880 C1OTW6 44579684 IC50 = 330 nM T32880 CE1KX7 44579685 IC50 = 400 nM T32880 CZF4B8 44579687 IC50 > 40000 nM T32880 C8A3XZ 44579730 IC50 = 2820 nM T32880 C6LQ9S 44579731 IC50 = 5540 nM T32880 CFN49B 44579732 IC50 = 66 nM T32880 CMI6G8 44579733 IC50 > 40000 nM T32880 CBVI46 44579734 IC50 = 730 nM T32880 CVD1W3 44591754 IC50 = 512 nM T32880 C3OL2Y 44591755 IC50 = 230000 nM T32880 C71GJA 44819566 IC50 > 400000 nM T32880 CKD8A7 44819735 IC50 > 400000 nM T32880 C1VH6I 45482712 IC50 = 78000 nM T32880 C0W6RQ 45482725 IC50 > 1000000 nM T32880 C34LSI 45482742 IC50 > 1000000 nM T32880 CK2R4F 45482768 IC50 > 1000000 nM T32880 CIU6F7 45482769 IC50 > 1000000 nM T32880 CJ7OS3 45482772 IC50 = 538000 nM T32880 CX42JP 45482778 IC50 > 1000000 nM T32880 C2HL7F 45486323 IC50 = 21 nM T32880 CUMF70 46899605 IC50 > 100000 nM T32880 C2DBN5 46899607 IC50 > 100000 nM T32880 C3G4QK 46899609 IC50 > 100000 nM T32880 CLK96Z 46899763 IC50 > 100000 nM T32880 CBOM64 46899765 IC50 > 100000 nM T32880 CA56RL 49831102 IC50 = 3 nM T32880 CU63QR 49847377 IC50 = 0.2 nM T32880 CZT4I8 49847378 IC50 = 0.2 nM T32880 CA72PE 49847379 IC50 = 1.6 nM T32880 CC23YW 49847498 IC50 = 55 nM T32880 CJ7H2B 49847753 IC50 = 3.4 nM T32880 C4V7EW 49848258 IC50 = 0.8 nM T32880 C4E2YF 49848485 IC50 = 13700 nM T32880 CWP7L0 49848519 IC50 = 427 nM T32880 CV0PU1 49848649 IC50 = 27 nM T32880 CP8TS6 49848895 IC50 = 0.4 nM T32880 C9COF5 49848896 IC50 = 0.5 nM T32880 CK0B1G 49848897 IC50 = 0.2 nM T32880 CP61VJ 49849002 IC50 = 0.2 nM T32880 C42SBF 49849005 IC50 = 4.3 nM T32880 CBM62Z 49849007 IC50 = 0.4 nM T32880 C05SEW 49849008 IC50 = 0.2 nM T32880 C78SAD 49849115 IC50 = 4.1 nM T32880 CF64IJ 49849120 IC50 = 0.2 nM T32880 CC9EB4 49849122 IC50 = 0.5 nM T32880 C2ORV5 49849123 IC50 = 5.4 nM T32880 CUJ4D6 49870967 IC50 = 100 nM T32880 CX8Z0D 50899320 IC50 = 120 nM T32880 C0HCX8 50916282 IC50 > 400000 nM T32880 C2QG8V 53318573 IC50 = 50118.72 nM T32880 C90UET 53319897 IC50 > 100000 nM T32880 CX7O4F 53319898 IC50 = 79432.82 nM T32880 CS3E2L 53493245 IC50 = 0.7 nM T32880 CRFI05 53493908 IC50 = 0.7 nM T32880 C68OFC 54681699 IC50 = 46 nM T32880 CJO04Q 54739165 IC50 < 50 nM T32880 CT0UM5 54741100 IC50 = 1.5 nM T32880 C28RDF 54746913 IC50 = 4.9 nM T32880 C35JDV 54746961 IC50 = 5.3 nM T32880 CDL06K 54746964 IC50 = 3.1 nM T32880 CK3GC9 54746970 IC50 < 10 nM T32880 C7Q4WV 54747815 IC50 < 10 nM T32880 C2TB1P 54747831 IC50 < 10 nM T32880 CZWR91 54747907 IC50 = 4.1 nM T32880 CT6MD1 54749350 IC50 = 0.65 nM T32880 C9OG0S 54749369 IC50 = 3 nM T32880 CU7S6Y 56656421 IC50 = 50 nM T32880 CMR1X3 56684140 IC50 > 1000000 nM T32880 CE26XI 56684141 IC50 > 1000000 nM T32880 CL8N7V 56964909 IC50 > 1000000 nM T32880 C34DJP 57384236 IC50 = 1.1 nM T32880 CEOC15 57384237 IC50 = 2 nM T32880 CY50WC 57384238 IC50 = 2.3 nM T32880 C7S0ZR 57384239 IC50 = 1.5 nM T32880 C2XN1G 57384481 IC50 = 1.6 nM T32880 CR73IZ 57384482 IC50 = 0.8 nM T32880 CR2M5H 57384483 IC50 = 0.5 nM T32880 CQ72HI 57384749 IC50 = 4.7 nM T32880 C68KGE 57384750 IC50 = 1.9 nM T32880 CA57BP 57384999 IC50 = 0.5012 nM T32880 C5OGF6 57385246 IC50 = 640 nM T32880 CJ8N5F 57385491 IC50 = 680 nM T32880 C2HXQ4 57385492 IC50 = 6600 nM T32880 CFB30C 57385493 IC50 = 2200 nM T32880 CE8A9F 57385494 IC50 = 1200 nM T32880 CHJ8G2 57385495 IC50 = 1000 nM T32880 CMSP14 57385496 IC50 = 7800 nM T32880 CB2Y1U 57385733 IC50 = 370 nM T32880 CH15PS 57385734 IC50 = 2600 nM T32880 CE40ZB 57385735 IC50 = 790 nM T32880 CKO54M 57385736 IC50 > 50000 nM T32880 C5XDF4 57385737 IC50 > 50000 nM T32880 CR7UN3 57385738 IC50 > 50000 nM T32880 C85XSW 57386006 IC50 > 50000 nM T32880 CUL23K 57386007 IC50 = 3040 nM T32880 CJTC03 57386008 IC50 = 440 nM T32880 C9THS0 57386009 IC50 = 15300 nM T32880 CV34YJ 57386010 IC50 > 50000 nM T32880 C0RKZ2 57386011 IC50 > 50000 nM T32880 COI01S 57386263 IC50 > 50000 nM T32880 CUF1Y0 57386264 IC50 = 3100 nM T32880 C2BJT0 57386265 IC50 = 840 nM T32880 CVZ19P 57386266 IC50 = 4700 nM T32880 C3SUV6 57386267 IC50 = 6000 nM T32880 CF0TG4 57386268 IC50 = 3.8 nM T32880 CCR1X8 57386520 IC50 = 98 nM T32880 CQ6JG3 57386521 IC50 = 31 nM T32880 CVK29R 57386523 IC50 = 2.1 nM T32880 C9S8MU 57386524 IC50 = 4.3 nM T32880 CMC8H6 57386782 IC50 = 0.4 nM T32880 CCT5D4 57386783 IC50 = 0.4 nM T32880 CC30XZ 57386784 IC50 = 5 nM T32880 C79BXP 57386785 IC50 = 0.8 nM T32880 CM6DV7 57387028 IC50 = 1 nM T32880 C0GS4F 57387282 IC50 = 0.6 nM T32880 C0TL9C 57387283 IC50 = 2.8 nM T32880 CRV2P5 57387539 IC50 = 0.2 nM T32880 CAU3G9 57387540 IC50 = 0.2 nM T32880 CL2AO8 57387541 IC50 = 0.4 nM T32880 C0XWL8 57387542 IC50 = 0.4 nM T32880 CC4DK0 57387775 IC50 = 1 nM T32880 C8DB9I 57387776 IC50 = 0.8 nM T32880 C2LZ8G 57387778 IC50 = 1200 nM T32880 CUN9V6 57388001 IC50 = 0.7 nM T32880 CV7W0P 57742961 IC50 = 65 nM T32880 CS6Z2D 57983461 IC50 < 100 nM T32880 C2DIK6 57983520 IC50 < 100 nM T32880 CCB65L 59603622 IC50 = 280 nM T32880 COL70Z 67049505 IC50 = 820 nM T32880 CKG14F 67049582 IC50 = 2500 nM T32880 CFM6H7 67049587 IC50 = 220 nM T32880 C3CU9D 67049655 IC50 = 7100 nM T32880 C7AJ1U 67049671 IC50 = 450 nM T32880 C2DPK9 67049808 EC50 = 4700 nM T32880 C3AP9U 67049854 IC50 = 1200 nM T32880 CB3HX6 67049905 IC50 = 1600 nM T32880 C5PM7A 67049973 EC50 = 14000 nM T32880 C4VG9Q 67050041 IC50 = 210 nM T32880 C6UHR9 67050359 IC50 = 730 nM T32880 C92WSG 67050361 EC50 = 13000 nM T32880 C7LBD8 67050367 IC50 = 850 nM T32880 C1N9OY 67050409 EC50 = 5800 nM T32880 C8VM6P 67283460 IC50 = 94 nM T32880 C5RGQ2 68392546 IC50 = 100 nM T32880 CKX41C 69674161 IC50 = 110 nM T32880 C4VU7J 70688210 IC50 = 4.9 nM T32880 CO7H3Q 71133989 IC50 = 2.3 nM T32880 CL3HT1 71449736 IC50 = 6300 nM T32880 CJH86V 71451542 IC50 > 100000 nM T32880 CH38AO 71453382 IC50 > 100000 nM T32880 C2U4AQ 71458738 IC50 = 14200 nM T32880 C1DYB4 71477196 IC50 = 17 nM T32880 C9XGE6 71537024 IC50 < 10 nM T32880 CK34XF 71538425 IC50 < 20 nM T32880 CX74LQ 71545631 IC50 = 18400 nM T32880 CP6WO8 71717922 IC50 = 20 nM T32880 C7Y8SB 71748680 IC50 = 15.85 nM T32880 CC7M4D 72204345 IC50 > 10000 nM T32880 CM41RB 72204346 IC50 > 10000 nM T32880 C9A4KH 72204347 IC50 > 10000 nM T32880 C5MZ7R 72204348 IC50 = 158.49 nM T32880 CA2C1U 72204349 IC50 = 199.53 nM T32880 C4JZ6C 72204350 IC50 = 794.33 nM T32880 CZFG12 72204539 IC50 = 630.96 nM T32880 C8PM1E 72204540 IC50 = 2.512 nM T32880 CT4X1K 72204541 IC50 = 1 nM T32880 CV4EJ6 72204542 IC50 = 79.43 nM T32880 C3X0TL 72204543 IC50 = 1995.26 nM T32880 CZF7R4 72204544 IC50 = 1258.93 nM T32880 CK63AC 72204738 IC50 = 3981.07 nM T32880 CGE63D 72204739 IC50 = 1000 nM T32880 CGR92Y 72204740 IC50 = 3162.28 nM T32880 CIBE51 72204741 IC50 = 398.11 nM T32880 C2C5QX 72204742 IC50 = 3162.28 nM T32880 C4JAC1 72204743 IC50 = 501.19 nM T32880 C3WV2R 72204920 IC50 = 1995.26 nM T32880 C4MO3I 72204921 IC50 = 630.96 nM T32880 C1E4BJ 72204922 IC50 = 7.943 nM T32880 CI0R2O 72204923 IC50 = 31.62 nM T32880 C40BFH 72204924 IC50 = 3.981 nM T32880 CB1G4W 72204925 IC50 = 25.12 nM T32880 C81AQS 72205106 IC50 = 39.81 nM T32880 CK5MI2 72205107 IC50 = 5.012 nM T32880 C35SGD 72205108 IC50 = 15.85 nM T32880 CI0ON6 72205109 IC50 = 50.12 nM T32880 C6LM0T 72205110 IC50 > 10000 nM T32880 CWJG76 72737642 IC50 = 14 nM T32880 C2UFG1 73052701 IC50 = 39 nM T32880 CW64KE 73052704 IC50 = 49 nM T32880 CZU9X4 73052863 IC50 = 13 nM T32880 C4XIZ8 73349624 IC50 = 12589.25 nM T32880 C68RKH 76310231 IC50 = 8500 nM T32880 C89AEL 76310612 IC50 = 0.7 nM T32880 CO1EN3 76317452 IC50 = 278000 nM T32880 CPE6U2 76335997 IC50 > 500000 nM T32880 C7K3JM 89812866 IC50 = 9400 nM T32880 CHVP04 92042841 IC50 = 61 nM T32880 C6NUD0 118718072 IC50 = 41800 nM T32880 CUR10H 118978237 IC50 = 5.8 nM T32880 CI5X2G 118978277 IC50 = 11 nM T32880 CH7WL3 118978299 IC50 = 20 nM T32880 C43IWX 118978308 IC50 = 22.9 nM T32880 C2LBH1 118978321 IC50 = 66 nM T32880 CB3I9Z 118978325 IC50 = 9 nM T32880 CWH4I0 118978339 IC50 = 19 nM T32880 C6XD3H 118978341 IC50 = 5.4 nM T32880 CJE6K4 118978367 IC50 = 7.3 nM T32880 CDBK07 118981498 IC50 = 2.6 nM T32880 CB23LS 118981525 IC50 = 10 nM T32880 C9F6RL 118981536 IC50 = 6.9 nM T32880 CF1E6T 118981546 IC50 = 6.8 nM T32880 C1ABC5 118981554 IC50 = 4.3 nM T32880 CR05OQ 118981555 IC50 = 4.2 nM T32880 CE9U5L 118981600 IC50 = 4 nM T32880 CO5XH7 118981638 IC50 = 4.9 nM T32880 CV84HB 118981731 IC50 = 4.4 nM T32880 CM3VL0 118981967 IC50 = 21 nM T32880 CW89CV 118982285 IC50 = 6.5 nM T32880 C51RST 121245332 IC50 = 3.8 nM T32880 C2LI6C 121245745 IC50 = 8.5 nM T32880 C69YAB 121246676 IC50 = 0.9 nM T32880 C27WIY 121246694 IC50 = 27 nM T32880 C0E7BZ 121246784 IC50 = 1.9 nM T32880 CH4O3R 121246791 IC50 = 1 nM T32880 C71YRT 121246805 IC50 = 5.4 nM T32880 CJU6X7 121246821 IC50 = 2 nM T32880 C1X3HT 121246837 IC50 = 6.1 nM T32880 C2UY6K 121246848 IC50 = 4.2 nM T32880 C5E0SB 121246859 IC50 = 1.8 nM T32880 CE3P9G 121246864 IC50 = 1.5 nM T32880 C6BIK2 121269752 IC50 = 0.62 nM T32880 C6H2YQ 122383780 IC50 = 96000 nM T32880 CT2UZ4 125377518 IC50 > 100000 nM T32880 C5NR3C 129027150 IC50 = 13700 nM T32880 CWO0V4 135566826 IC50 = 2800 nM T32880 CV9J3Z 135737442 IC50 = 195000 nM T32880 CSCH32 135871166 IC50 = 27500 nM T32880 C3Q9KJ 135871167 IC50 = 81000 nM T32880 CJIK12 135871172 IC50 = 2200 nM T32880 CWI9V2 135871182 IC50 = 2100 nM T32880 C39VQA 135871218 IC50 = 700 nM T32880 CF5TV8 135871220 IC50 = 3800 nM T32880 CD6QM3 135871221 IC50 = 800 nM T32880 C2G7XC 135871222 IC50 = 24000 nM T32880 CAJ08Y 135871235 IC50 = 400 nM T32880 C42ISC 135871238 IC50 = 1400 nM T32880 C9DPJ0 135871283 IC50 = 2000 nM T32880 CYVH90 135895253 IC50 = 8 nM T32880 CT57ZH 136069450 IC50 = 0.2 nM T32880 CFT9R3 136069453 IC50 = 0.6 nM T32880 CRPQ42 136069494 IC50 = 2.5 nM T32880 CK8Z3V 136069521 IC50 = 5 nM T32880 CPY1B2 136069522 IC50 = 31 nM T32880 CX0OM4 136069523 IC50 = 11 nM T32880 C6EU4D 136069524 IC50 = 76 nM T32880 CQA2Z1 136069531 IC50 = 9.3 nM T32880 CCH31A 136069532 IC50 = 0.9 nM T32880 CH8GV7 136069561 IC50 = 14 nM T32880 CQ1FS4 136069563 IC50 = 3.9 nM T32880 C97REI 136074309 IC50 = 6000 nM T32880 CN6X7E 136074310 IC50 = 13500 nM T32880 CLV1R6 136074312 IC50 = 5700 nM T32880 CY3Z2V 136074313 IC50 = 1200 nM T32880 CEJ1M9 136074314 IC50 = 3000 nM T32880 CR5IM8 136074315 IC50 = 3400 nM T32880 CX02WY 136074316 IC50 = 2400 nM T32880 CICS75 136074317 IC50 = 7300 nM T32880 CS9C0Q 136074318 IC50 = 3900 nM T32880 CQTB32 136205798 IC50 = 1.1 nM T32880 CV8QP3 136205832 IC50 = 0.2 nM T32880 CB93EM 136205833 IC50 = 0.6 nM T32880 CV1C5I 136986966 IC50 = 2600 nM T32880 CJNU29 137083353 IC50 = 12 nM T32880 C0F8XB 137150345 IC50 = 20 nM T32880 C5UFR2 138319689 IC50 = 62.23 nM T32880 C7RYB5 141508724 IC50 = 248 nM T32880 CI1DE9 141508725 IC50 = 280.6 nM T32880 C5PN8T 141508727 IC50 = 228.2 nM T32880 CE36KV 141508729 IC50 = 418.3 nM T32880 C29GLS 141508732 IC50 = 278.3 nM T32880 C8SW9L 141508738 IC50 = 75.82 nM T32880 C5NJS7 141508739 IC50 = 61.08 nM T32880 C0Q5YG 141508741 IC50 = 308.3 nM T32880 C4QT0G 141508742 IC50 = 759.4 nM T32880 C2XB9I 141508745 IC50 = 418.7 nM T32880 CLK1B4 141508746 IC50 = 419.3 nM T32880 CJ9O3L 141508747 IC50 = 77 nM T32880 CV6N8B 141508748 IC50 = 271 nM T32880 C5SIU2 141508749 IC50 = 67.58 nM T32880 C2JRM3 141508751 IC50 = 231.1 nM T32880 C3WIL6 141508752 IC50 = 375.4 nM T32880 CK2ST8 141508755 IC50 = 418.3 nM T32880 CG0FL4 141508765 IC50 = 52.84 nM T32880 CN8EK0 141508769 IC50 = 579.7 nM T32880 CVMW03 141617793 EC50 = 17000 nM T32880 C2ML4K 141740991 IC50 = 1.9 nM T32880 C15DMN 145955244 IC50 = 16000 nM T32880 CK41QM 145957905 IC50 = 650 nM T32880 CWU6S2 145958372 IC50 = 6500 nM T32880 C7SIP1 145960425 IC50 = 801.4 nM T32880 CID5Y8 145960662 IC50 = 2165 nM T32880 CC9A8D 145960865 IC50 = 3594 nM T32880 CZDC15 145961128 IC50 = 853.8 nM T32880 CVZ8E9 145961326 IC50 = 3086 nM T32880 CEJ90L 145961795 IC50 = 853.8 nM T32880 C9R1SO 145961819 IC50 = 69 nM T32880 CB62WJ 145961830 IC50 = 6995 nM T32880 C4C6NP 145962038 IC50 = 995.8 nM T32880 C2Y7SM 145962118 IC50 = 1507 nM T32880 C6D5GL 145962572 IC50 = 608.2 nM T32880 CPO03J 145962836 IC50 = 5527 nM T32880 CJS57A 145962965 IC50 = 2291 nM T32880 C6YJ5R 155539215 IC50 = 905 nM T32880 COL30E 155540589 IC50 = 63 nM T32880 C5MFJ8 155548449 IC50 = 143 nM T32880 CN7H9B 155554391 IC50 = 70 nM T32880 C0GU8Y 155559177 IC50 > 25000 nM T32880 CG7R3L 155559901 IC50 = 4.8 nM T32880 CGU0A2 155563031 IC50 > 25000 nM T32880 C32NYC 155565735 IC50 > 25000 nM T32880 D07IOY 10365 IC50 = 6100 nM T32880 D08IZY 3080614 Ki = 8000 nM T32880 D08JSE 45102710 IC50 = 100 nM T32880 D0B2WZ 15331 IC50 > 100000 nM T32880 D0R6GQ 1198 IC50 > 10000000 nM T32880 D0WA3E 54685215 IC50 = 22 nM T32880 D0X5US 459617 IC50 = 15000 nM T51487 D02YPG 667484 EC50 = 11000 nM T51487 D06ZII 969472 Ki = 50.1 nM T51487 D07JVL 3016 Ki = 16 nM T51487 D0D5GD 3373 Ki = 3.3 nM T51487 D0F0YZ 4737 IC50 = 1000000 nM T51487 D0L9GG 2118 EC50 = 37 nM T51487 D0T1WN 5732 IC50 = 14 nM T51487 D0A5MC 11712649 IC50 = 330 nM T51487 D0CH7C 57336276 Ki = 985 nM T51487 D0HO2T 23581869 Ki = 0.5 nM T51487 D0S4JK 24771867 IC50 = 490 nM T51487 D0Z9HW 23630026 Ki = 0.5 nM T51487 C7SZ9E 613843 IC50 > 10000 nM T51487 C12NWX 2729103 IC50 > 10000 nM T51487 CO61AF 2820320 IC50 > 10000 nM T51487 C59BWK 2820473 IC50 = 470 nM T51487 C1Z6YU 9821389 Ki = 71 nM T51487 CCX58U 9865233 Ki = 0.73 nM T51487 C1VRB9 9951530 EC50 = 56 nM T51487 CPC3U1 9971547 Ki = 362 nM T51487 CUT5W8 9976743 EC50 = 53 nM T51487 CUSM85 10221761 Ki = 1.3 nM T51487 CBQ4R7 10905261 EC50 = 36 nM T51487 C15NXT 10926766 EC50 = 266 nM T51487 CK1S7J 10927005 EC50 = 107 nM T51487 CWK02D 10936672 EC50 = 135 nM T51487 C09PCZ 10971225 EC50 = 92 nM T51487 CG9Z6N 10991911 EC50 = 17 nM T51487 C7DVK8 11014215 EC50 = 120 nM T51487 CJB1V2 11035207 EC50 = 258 nM T51487 C31EGD 11036467 EC50 = 81 nM T51487 CBV36I 11047145 EC50 = 127 nM T51487 C8B7TF 11067772 EC50 = 95 nM T51487 CNSA17 11143256 EC50 = 136 nM T51487 CCU8G9 11526006 IC50 = 150 nM T51487 CWO70Q 11673720 Ki = 15 nM T51487 CX7G9K 11759134 EC50 = 170 nM T51487 CL4XD0 11783674 EC50 = 18 nM T51487 CB9U0F 11825216 EC50 = 28 nM T51487 CTI32Y 15680235 EC50 < 100 nM T51487 C8SR4O 25187292 IC50 = 46 nM T51487 C6DBS4 25187295 IC50 = 50 nM T51487 CF1B8A 25188671 IC50 = 50 nM T51487 CW97NA 44273000 IC50 = 1 nM T51487 C5KV7A 44364531 EC50 = 208 nM T51487 CZK75V 44364548 EC50 = 118 nM T51487 C0FN6W 44364725 EC50 = 2200 nM T51487 CYE1R8 44364726 EC50 = 41 nM T51487 CE8F3Y 44364734 EC50 = 303 nM T51487 COH5G6 44364735 EC50 = 544 nM T51487 C2VHW7 44364747 EC50 = 133 nM T51487 CZL2P0 44364907 EC50 = 69 nM T51487 CCX08E 44364918 EC50 = 93 nM T51487 C6D3BI 44560284 EC50 = 250 nM T51487 C6J0GP 44561356 IC50 = 580 nM T51487 C9UW4V 44561357 IC50 = 580 nM T51487 CZR6A5 44561358 IC50 > 10000 nM T51487 C4IF7B 44561386 IC50 = 1000 nM T51487 C3GZU0 44576235 EC50 = 11000 nM T51487 C63IYQ 51003493 IC50 = 134 nM T51487 CP8IG3 53317278 IC50 = 64 nM T51487 CP9I6O 53319883 IC50 = 74 nM T51487 CO6P3V 53320033 IC50 = 242 nM T51487 CCZ98L 53321188 IC50 = 67 nM T51487 C8MZR1 53322513 IC50 = 157 nM T51487 CTG2S9 53322514 IC50 > 3000 nM T51487 C29ARN 53323855 IC50 = 1 nM T51487 CBGD06 53323856 IC50 = 94 nM T51487 C9DJP1 53326435 IC50 = 64 nM T51487 CBO9L1 60194848 IC50 = 120000 nM T51487 CU83BZ 60194849 IC50 = 3800 nM T51487 CQ91VU 118278442 Ki = 140 nM T51487 CH0D4J 130439777 Ki = 850 nM T51487 C56XBU 130439778 Ki = 55000 nM T51487 C9N8LW 130439889 Ki = 542 nM T51487 C89LNZ 136118605 IC50 = 479 nM T51487 D06SOQ 6918451 Ki = 0.88 nM T51487 D09IHE 6918583 Ki = 0.8 nM T51487 D0E7PY 11624499 Ki = 174 nM T51487 D0M4CP 5081 EC50 = 1.1 nM T51487 D0O9MG 5311203 Ki = 17 nM T52921 D04CRN 54841 IC50 > 5000 nM T52921 D0CS2F 3955 Ki > 10000 nM T52921 D0PG8O 5360515 Ki > 10000 nM T52921 D0U5FS 3396 Ki = 500 nM T52921 D03TBJ 11848225 Ki = 0.9 nM T52921 D0G2XE 6918468 IC50 = 2200 nM T52921 D0W4YO 16131448 Ki = 0.04898 nM T52921 D0M1YN 5311194 Ki = 0.403 nM T52921 D00ACC 9844019 Ki = 1.12 nM T52921 D08AWI 11430856 Ki > 2000 nM T52921 CBGO28 70419 Ki = 11 nM T52921 C3HB4V 416359 IC50 = 200 nM T52921 CQ6MW0 3655995 EC50 = 174 nM T52921 CLW4B1 5311340 Ki = 8.2 nM T52921 CD49UV 9797246 Ki = 133 nM T52921 CNO0W4 9799433 Ki = 5.22 nM T52921 CYR3O0 9802205 Ki = 50.7 nM T52921 CPG57N 9803475 Ki = 12.9 nM T52921 CX7DO4 9806799 Ki = 4.05 nM T52921 CK6GR9 9816910 IC50 > 5000 nM T52921 CE6NF9 9823363 IC50 = 1.3 nM T52921 C6LGX9 9824268 Ki = 82.4 nM T52921 C7TDX2 9824313 Ki = 46.7 nM T52921 C70KEP 9824565 Ki = 0.5 nM T52921 C06LIG 9825723 Ki = 2.3 nM T52921 CPK4X7 9836463 Ki = 1054 nM T52921 C6Y7NA 9844540 Ki = 2 nM T52921 C0F9RX 9845765 Ki = 7 nM T52921 C8M4HT 9846747 Ki = 2.2 nM T52921 CE2YQ9 9848110 Ki = 2 nM T52921 CKD2H4 9848990 Ki = 77 nM T52921 CLQ6Z8 9866158 Ki = 0.5 nM T52921 CEO0M2 9880173 Ki = 414 nM T52921 CPYK08 9887195 IC50 = 820 nM T52921 CV2G7M 9889948 Ki = 11.8 nM T52921 C1VM4H 9902583 Ki = 692 nM T52921 C5BC4P 9902874 Ki = 39 nM T52921 CX3CM8 9905428 Ki = 1.39 nM T52921 C2TE5X 9922658 Ki = 10 nM T52921 C4NJ0W 9923726 Ki = 125 nM T52921 CIUE54 9924406 Ki = 5.4 nM T52921 C5HN0J 9925137 Ki = 1.1 nM T52921 CZT2J0 9927928 Ki = 18.66 nM T52921 C2U8XH 9932834 Ki = 3.4 nM T52921 C9MK3B 9934232 Ki = 6.8 nM T52921 CUBQ95 9937777 Ki = 2.25 nM T52921 C4FD7V 9947044 Ki = 1.4 nM T52921 CG9ER5 9947155 Ki = 2297 nM T52921 COFT18 9951673 Ki = 4 nM T52921 C3GXH0 9954388 Ki = 5.6 nM T52921 CT8C2X 9958643 Ki = 1.8 nM T52921 CE3CJ4 9969865 Ki = 5102 nM T52921 CAGL19 9997843 Ki = 0.7 nM T52921 CL9QS0 10004950 IC50 = 19 nM T52921 C4N8YE 10020165 Ki = 6 nM T52921 C25DYT 10022859 Ki = 0.52 nM T52921 CFOK60 10042904 Ki = 3.96 nM T52921 CC60VS 10052051 Ki = 505 nM T52921 CV1OU6 10109140 Ki = 4.4 nM T52921 C7YCF1 10109899 Ki = 1 nM T52921 CJNE19 10110916 Ki = 225 nM T52921 C76MVA 10111186 Ki > 10000 nM T52921 CWEC34 10114637 Ki = 4461 nM T52921 C40BMF 10133108 Ki = 51 nM T52921 C2WZ9G 10133332 Ki = 1259 nM T52921 CP1SO7 10134077 Ki = 11 nM T52921 CEG0M4 10134217 Ki = 357 nM T52921 C3ZTU0 10137134 Ki = 225 nM T52921 C83KDV 10137876 Ki = 7.4 nM T52921 C8E9KP 10139672 Ki = 41 nM T52921 CQGE97 10150001 Ki = 94 nM T52921 C76SOW 10150260 Ki = 37 nM T52921 CRC46J 10154739 Ki = 634 nM T52921 CKN3A8 10154848 Ki = 410 nM T52921 CFIL01 10155966 Ki = 2.3 nM T52921 CIO6U3 10156336 Ki = 1239 nM T52921 CP53IB 10156591 Ki = 0.4 nM T52921 CI1U4Z 10156821 Ki = 7.5 nM T52921 CTO0N5 10158555 Ki = 31 nM T52921 CG51TX 10159203 Ki = 11 nM T52921 CWM2X6 10160920 Ki = 18 nM T52921 CB57JZ 10171862 Ki = 78 nM T52921 CDV15J 10172398 Ki = 58 nM T52921 CJN21A 10178311 Ki = 184 nM T52921 CHN4G6 10178563 Ki = 824 nM T52921 C5RO6K 10182346 Ki = 7114 nM T52921 CNZL85 10193971 Ki = 347 nM T52921 CN79QX 10194236 Ki = 31 nM T52921 CWC8L1 10199945 IC50 = 2.5 nM T52921 C12NGT 10199984 Ki = 3454 nM T52921 CH40KY 10202108 Ki = 437 nM T52921 CV1T7R 10202241 Ki > 10000 nM T52921 CYB0H9 10221539 IC50 = 3.3 nM T52921 CM27FK 10225083 Ki = 2 nM T52921 CZ0C5T 10252647 Ki = 66 nM T52921 CH54KF 10260917 EC50 = 0.1585 nM T52921 C8PL7B 10274330 Ki = 33 nM T52921 CR1HX2 10275388 Ki = 4358 nM T52921 CSO8D7 10276738 Ki = 0.38 nM T52921 CDP01X 10286440 Ki = 570 nM T52921 C1FE9H 10286996 Ki = 105 nM T52921 CJ14VU 10291377 Ki = 16 nM T52921 C61OKS 10292091 Ki = 111 nM T52921 CV0T3H 10301207 Ki = 1 nM T52921 C1ENR2 10323169 Ki = 2.3 nM T52921 CD09RQ 10338496 Ki = 110 nM T52921 C0G7RF 10362733 Ki = 4544 nM T52921 C59JAP 10363496 Ki = 2.2 nM T52921 CAYF18 10385808 Ki = 2.6 nM T52921 C95EWP 10395965 Ki = 27 nM T52921 CWK4O1 10406239 Ki = 0.1 nM T52921 CTA8Q0 10407144 Ki = 19.6 nM T52921 CX4TS2 10413540 Ki = 78 nM T52921 CYHC38 10430819 Ki = 0.5495 nM T52921 CZP0C7 10441529 EC50 = 0.302 nM T52921 CZ6I9V 10451761 IC50 = 6.8 nM T52921 CKMN08 10475466 Ki = 4.6 nM T52921 C1DI7F 10500922 Ki = 218 nM T52921 C90DEM 10504545 Ki = 6.8 nM T52921 CDK8W2 10548749 Ki = 5.8 nM T52921 C54EOA 10572810 Ki = 7.3 nM T52921 CD9JB5 10574643 Ki = 2.8 nM T52921 CQ74CO 10593778 Ki = 2.5 nM T52921 CZQ4J6 10596013 Ki = 79.9 nM T52921 CHV5D1 10601891 Ki = 15 nM T52921 CS84IW 10618605 Ki = 2.5 nM T52921 CPC52U 10646744 Ki = 7.2 nM T52921 C10KTE 10646745 Ki = 8.5 nM T52921 CH16SQ 10668903 Ki = 85.6 nM T52921 CMT48G 10669669 Ki = 20.4 nM T52921 CF7SX5 10669670 Ki = 13.2 nM T52921 CP25HJ 10669671 Ki = 37.3 nM T52921 CHC1I4 10697286 Ki = 15.3 nM T52921 C2RN9F 10713623 Ki = 10.2 nM T52921 C8XB3K 10714523 Ki = 1.4 nM T52921 CY36JZ 10715725 Ki = 88.5 nM T52921 CFH5N0 10715726 Ki = 121.2 nM T52921 C48PSE 10718869 Ki = 2.6 nM T52921 CN05WO 10763594 Ki = 0.39 nM T52921 CBC6U3 10765154 Ki = 1.8 nM T52921 CXF9R4 10766007 Ki = 1.8 nM T52921 CDJP34 10783436 IC50 = 6.8 nM T52921 CTR2I0 10788833 Ki = 6.5 nM T52921 CQS8K6 10789513 Ki = 1.8 nM T52921 C9SN6H 10831914 Ki = 369.3 nM T52921 CS3Y4G 10832076 IC50 = 5.9 nM T52921 CMVI50 10832445 Ki = 6.3 nM T52921 CPG23C 10836379 Ki = 20.7 nM T52921 C4IT2B 10837001 Ki = 3.3 nM T52921 C2QIL3 10876990 EC50 = 1 nM T52921 CWJL70 10905740 IC50 = 434 nM T52921 C4TSV6 10927662 Ki = 0.5248 nM T52921 C1TSN4 10928037 Ki = 0.7762 nM T52921 CT5UO7 10937810 Ki = 2.188 nM T52921 CU09AV 10937901 IC50 = 38 nM T52921 CVP6D3 10942284 EC50 = 0.2692 nM T52921 CN7XS4 10948527 IC50 = 340 nM T52921 CSLT97 10949380 IC50 = 283 nM T52921 C9FYG3 10950562 Ki = 1.66 nM T52921 CHK23I 10961428 Ki = 1.66 nM T52921 C2HP7F 10981761 IC50 = 758 nM T52921 C78FTE 10986100 EC50 = 63.1 nM T52921 C8Q6YE 11004121 Ki = 0.4467 nM T52921 CIR4E5 11007758 EC50 = 134.9 nM T52921 C0R2DW 11007770 EC50 = 31.62 nM T52921 C3V7LT 11014751 Ki = 0.6457 nM T52921 CY0S2I 11029698 EC50 = 257.04 nM T52921 CRP95V 11051525 EC50 = 0.2512 nM T52921 C9Z7BY 11115933 EC50 = 1.413 nM T52921 CDU0E5 11123873 Ki = 2.089 nM T52921 CU6PV0 11143820 IC50 = 97 nM T52921 C7HM0O 11152739 Ki = 3.5 nM T52921 C26ENL 11164004 Ki = 15.6 nM T52921 C62WBJ 11165726 Ki = 135 nM T52921 C4COM2 11170657 Ki = 0.05 nM T52921 C3TW2O 11187225 Ki = 4.5 nM T52921 C6EWJ9 11188910 Ki = 4.4 nM T52921 CUBX19 11189444 IC50 > 10000 nM T52921 CTKF50 11191683 IC50 = 5.5 nM T52921 CS5ET8 11212373 IC50 > 10000 nM T52921 C26MVG 11223982 IC50 > 10000 nM T52921 C4QT5Y 11233481 Ki = 15.5 nM T52921 CW1O5V 11256620 Ki = 12 nM T52921 CPBZ36 11274537 Ki > 5000 nM T52921 C4FRH7 11315651 Ki = 1.64 nM T52921 C5DBK1 11326750 Ki = 11 nM T52921 CJM7R5 11327115 Ki = 253 nM T52921 CW7SN4 11329662 Ki = 0.5012 nM T52921 CS1W7V 11338717 IC50 > 10000 nM T52921 CY0SV8 11349939 Ki > 10000 nM T52921 C6UZF7 11371415 Ki = 11.7 nM T52921 C4BZ1C 11372427 Ki = 4.3 nM T52921 CQC4G5 11372671 IC50 = 6150 nM T52921 CT6Z0B 11393860 Ki = 29.3 nM T52921 CGO58L 11406629 IC50 = 3700 nM T52921 CBJ0X5 11407510 IC50 > 10000 nM T52921 CU5GO6 11411841 IC50 = 25.2 nM T52921 CW0E4L 11418847 IC50 > 10000 nM T52921 C9KV1U 11451023 Ki = 5.64 nM T52921 C7UDE8 11461888 Ki = 7.49 nM T52921 CF6DQ2 11462727 Ki = 10 nM T52921 CKIQ83 11463791 IC50 > 10000 nM T52921 CC9TX5 11464294 IC50 > 10000 nM T52921 CMU9K5 11464846 Ki = 0.336 nM T52921 C3BA5F 11480038 Ki = 72 nM T52921 CVQ70S 11480201 Ki = 0.04 nM T52921 C41MEV 11511090 IC50 = 0.22 nM T52921 CZ4OM7 11516508 Ki = 2.2 nM T52921 C2N3BS 11523928 IC50 > 1000 nM T52921 CJE45X 11523929 IC50 > 1000 nM T52921 CL1O0H 11523972 IC50 = 350 nM T52921 CQ30PM 11525624 IC50 = 42 nM T52921 C8TZ9G 11544654 IC50 = 32 nM T52921 CS0B4G 11544795 Ki = 2.4 nM T52921 C3DG8U 11552010 Ki = 10.2 nM T52921 C10BUF 11559590 IC50 > 1000 nM T52921 C5ZR9W 11559820 IC50 = 540 nM T52921 CG6UM9 11561261 IC50 > 1000 nM T52921 CRX48F 11581029 Ki = 18.9 nM T52921 CA35LD 11583008 Ki = 4.6 nM T52921 CVA8L6 11583016 IC50 = 4 nM T52921 C1WBQ5 11597677 IC50 = 83 nM T52921 CY72UC 11602409 Ki = 8.5 nM T52921 C0AOU4 11603249 IC50 = 730 nM T52921 C38FTP 11619363 IC50 = 12 nM T52921 C8RKH0 11619553 IC50 = 8.3 nM T52921 C9WMX4 11624970 Ki = 29.8 nM T52921 C34OQC 11626062 Ki = 1.74 nM T52921 CF6R4S 11632761 IC50 > 1000 nM T52921 C4ZD1X 11633324 IC50 = 7.5 nM T52921 CIY0O4 11639705 IC50 > 1000 nM T52921 CFV5Q1 11661648 IC50 > 1000 nM T52921 CPN46U 11676849 IC50 = 580 nM T52921 C4ULQ7 11710187 IC50 = 23 nM T52921 CE0D1U 11743914 Ki = 116 nM T52921 CV8CF3 11749578 IC50 > 10000 nM T52921 CFRY36 11757207 Ki = 15 nM T52921 CED7I5 11761926 Ki = 0.6607 nM T52921 CCY92E 11768467 EC50 = 7.244 nM T52921 CG9HW8 11795019 Ki = 2.9 nM T52921 CN9M8E 11811722 IC50 = 2420 nM T52921 C8UE5W 11826819 Ki = 2.138 nM T52921 CS7W2V 11848793 Ki = 1.7 nM T52921 CJ34HP 11956520 Ki = 0.19 nM T52921 CA5ZX7 11956918 Ki = 9.4 nM T52921 C14RWU 11967729 EC50 = 10.96 nM T52921 CP1AZ0 11967746 EC50 = 26.3 nM T52921 CF01LM 12986253 Ki = 1.9 nM T52921 C63ASY 12986256 Ki = 120 nM T52921 CAW1M2 15512228 Ki = 0.52 nM T52921 C30CHU 15512229 Ki = 0.2512 nM T52921 C9B5OD 15512233 Ki = 39.81 nM T52921 CX6H8V 15512234 Ki = 1.259 nM T52921 CC5X0L 15512235 Ki = 3.981 nM T52921 CG0CS6 15512236 Ki = 15.85 nM T52921 C53KRM 15512237 Ki = 0.3162 nM T52921 CLA5K8 15512238 Ki = 3.981 nM T52921 C4I5TU 15512239 Ki = 10 nM T52921 CSX74V 15512240 Ki = 1.585 nM T52921 CET25R 15512241 Ki = 5.012 nM T52921 C23GHP 15512242 Ki = 100 nM T52921 C7CNY1 15512243 Ki = 1.585 nM T52921 CZA4J8 15541261 Ki = 23 nM T52921 CE18TP 15586319 Ki = 810 nM T52921 CD7K0Y 15965865 IC50 = 6000 nM T52921 CHN45W 15982524 IC50 = 510 nM T52921 CRX3U8 15982526 IC50 = 680 nM T52921 C6DW5M 15982528 IC50 > 10000 nM T52921 C7Z8OD 15982529 IC50 = 7400 nM T52921 CHO67K 15982530 IC50 = 600 nM T52921 C3B8AG 15982657 IC50 = 880 nM T52921 C4W6CK 15982658 IC50 = 140 nM T52921 CLWI08 15982659 IC50 = 10000 nM T52921 CV1G7O 15982660 IC50 = 83 nM T52921 CG3L8Z 15982661 IC50 = 120 nM T52921 CN64AP 15982791 IC50 = 320 nM T52921 C7KXO3 15982794 IC50 > 10000 nM T52921 CB1CR0 15982795 IC50 = 100 nM T52921 C0PKF1 15982796 IC50 = 10000 nM T52921 C3HL5F 15982797 IC50 = 820 nM T52921 CJY21D 15982932 IC50 > 10000 nM T52921 CJ6W1T 15982933 IC50 < 10000 nM T52921 CK97VS 15982935 IC50 = 250 nM T52921 C8TQ4B 15982937 IC50 = 900 nM T52921 C1PB8H 15982938 IC50 = 1120 nM T52921 CS46QG 15983062 IC50 = 800 nM T52921 CXJ61F 15983063 IC50 = 3600 nM T52921 CIG32A 15983065 IC50 = 10000 nM T52921 CG96OQ 15983067 IC50 = 2750 nM T52921 CA5GL7 16007142 Ki = 4 nM T52921 CDR71P 16043240 IC50 > 10000 nM T52921 C4H2NO 16061455 Ki = 6 nM T52921 C08RXS 16665915 Ki = 800 nM T52921 CS9FW1 16665917 Ki = 290 nM T52921 C1LX0I 16665918 Ki = 18 nM T52921 C6W9BJ 16733371 Ki = 6 nM T52921 C4ORI6 16739256 Ki = 15.1 nM T52921 C1MFJ2 16747695 Ki = 4.1 nM T52921 CG84KV 17858339 IC50 = 320 nM T52921 CWXD07 17858448 IC50 = 4.7 nM T52921 C8AZW7 18441735 IC50 = 15000 nM T52921 C1Y9FT 18782352 Ki = 0.9 nM T52921 CYUG80 18782376 Ki = 10.8 nM T52921 C46DPT 18782378 Ki = 2 nM T52921 C73DWV 18782384 Ki = 14.5 nM T52921 CHAI36 22272877 IC50 = 17 nM T52921 C5VSD6 22272900 IC50 = 17 nM T52921 CB5DY1 22272974 IC50 = 3.9 nM T52921 C1NU9M 22273044 IC50 = 2.1 nM T52921 CX3JY4 22273116 IC50 = 120 nM T52921 CRZ72H 22273255 IC50 = 3100 nM T52921 C8DF5U 22558157 Ki = 12 nM T52921 C1R5PV 22562132 Ki = 5670 nM T52921 CJ8OB0 22562135 Ki = 3592 nM T52921 C0GKU4 22562137 Ki = 20.4 nM T52921 CJ86RS 22725091 Ki = 10 nM T52921 CL7X2U 23383556 Ki = 0.4 nM T52921 COHN67 23383564 Ki = 0.5 nM T52921 C46ZSX 23542099 IC50 = 34 nM T52921 CVLY78 23542106 IC50 = 82 nM T52921 CB9MC8 24735827 Ki = 119 nM T52921 CWP85S 24776395 Ki = 3.1 nM T52921 CVD48X 24776396 Ki = 186 nM T52921 C3WDL8 24776397 Ki = 8.9 nM T52921 CXL4R0 24776398 Ki = 21 nM T52921 CR9I1S 24776399 Ki = 395 nM T52921 CQDJ35 24776400 Ki = 147 nM T52921 C6CX0Z 24776401 Ki = 6.6 nM T52921 CJH18I 24776402 Ki = 12 nM T52921 C27SGI 24776403 Ki = 26 nM T52921 CV5IG2 24776404 Ki = 51 nM T52921 CQ70IW 24776405 Ki = 81 nM T52921 CQ2P5J 24776406 Ki = 136 nM T52921 CYIV42 24776407 Ki = 4.7 nM T52921 CWB06Z 24776408 Ki = 23 nM T52921 C36WQO 24776409 Ki = 42 nM T52921 CUP2C6 24776410 Ki = 90 nM T52921 CC3W7E 24776411 Ki = 130 nM T52921 C3N6GE 24776412 Ki = 65 nM T52921 C2M6BR 24776413 Ki = 92 nM T52921 C8SXV9 24799146 Ki = 180 nM T52921 C1S2NC 24799325 Ki = 104 nM T52921 CLAU56 24799509 Ki = 100 nM T52921 C2VHP0 24799848 Ki = 545 nM T52921 C26ZYM 24800015 Ki = 260 nM T52921 CWV5F4 24800016 Ki = 740 nM T52921 CS01RL 24800107 Ki = 2.1 nM T52921 CL2WB0 24800108 Ki = 0.0858 nM T52921 CY89FP 24800188 Ki = 186 nM T52921 C13MJI 24822630 EC50 = 0.1 nM T52921 C6TWH4 24824635 EC50 = 88 nM T52921 CYM02E 24847114 IC50 = 15 nM T52921 C9O5NZ 24857819 IC50 = 0.65 nM T52921 CN0T1F 24857820 IC50 = 0.66 nM T52921 CS5D1K 24882570 IC50 = 0.033 nM T52921 CQ63PM 24894425 Ki = 17 nM T52921 C2EQR6 24894426 Ki = 0.47 nM T52921 CT9EZ4 24894428 Ki = 1.1 nM T52921 CN1E8M 24894430 Ki = 30 nM T52921 C9USO6 24894431 Ki = 58 nM T52921 C4IDR3 24894531 Ki = 11 nM T52921 CA8E4J 24894533 Ki = 21 nM T52921 C2AU5Y 24894647 Ki = 20 nM T52921 C8JL9I 24894652 Ki = 49 nM T52921 C6AZ9P 24894653 Ki = 25 nM T52921 CC6F9D 24894783 Ki = 51 nM T52921 CDLW86 25001412 Ki = 0.7244 nM T52921 CBIU48 25077447 EC50 = 4.37 nM T52921 CFB8G1 25077910 EC50 = 25 nM T52921 CHWB32 25082025 EC50 = 156 nM T52921 C2FPI9 25084159 EC50 = 22.3 nM T52921 C6HL3Q 25089553 EC50 = 0.1349 nM T52921 CP56DF 25089995 IC50 = 0.471 nM T52921 CF6RA5 25190572 Ki = 84 nM T52921 CPK5D7 25190573 Ki = 34 nM T52921 CON62K 25190574 Ki = 57 nM T52921 C6S3WN 25190575 Ki = 83 nM T52921 CF15AH 25190576 Ki = 53 nM T52921 CBN1Q0 25190577 Ki = 89 nM T52921 CKB72D 25190578 Ki = 234 nM T52921 CZR78G 25190579 Ki = 203 nM T52921 CF2JK0 25190580 Ki = 48.7 nM T52921 CE4R2X 25190581 Ki = 56 nM T52921 CYC6S0 25190582 Ki = 19.5 nM T52921 CE61QB 25190583 Ki = 18.5 nM T52921 C9V8MS 25190584 Ki = 26 nM T52921 C3UV5M 25190585 Ki = 47.8 nM T52921 CKFI42 25190586 Ki = 2.1 nM T52921 C5UQX3 25190587 Ki = 2.55 nM T52921 C5J2WE 25190588 Ki = 8.65 nM T52921 CX84WI 25190589 Ki = 5 nM T52921 C5RUI9 25190590 Ki = 3.5 nM T52921 CQY69C 25190591 Ki = 3.7 nM T52921 C8SEQ2 25190592 Ki = 12.1 nM T52921 C5BS7N 25190593 Ki = 2.15 nM T52921 CE19OU 25190594 Ki = 2.75 nM T52921 CP5ID6 25190595 Ki = 3.8 nM T52921 CO8E4G 25190596 Ki = 3.2 nM T52921 CX87HD 25190597 Ki = 8 nM T52921 CY6CV1 25190598 Ki = 2.3 nM T52921 CW5UP9 25190599 Ki = 0.8 nM T52921 C1C8VK 25190600 Ki = 0.7 nM T52921 CL7Q2F 25190601 Ki = 0.7 nM T52921 CD0H5U 25190602 Ki = 0.5 nM T52921 C8OWC0 25190603 Ki = 0.5 nM T52921 CH06YU 25190604 Ki = 0.6 nM T52921 CEJ25L 25190605 Ki = 0.5 nM T52921 CXD5R8 25190606 Ki = 1 nM T52921 CU6W8O 25190607 Ki = 5.4 nM T52921 CWJB54 25190608 Ki = 4.5 nM T52921 CMHS48 25190609 Ki = 1.7 nM T52921 CBL9S4 25190610 Ki = 2.1 nM T52921 CZ8Y6L 25190611 Ki = 1.6 nM T52921 CL9SN6 25190612 Ki = 1.4 nM T52921 C1MGY3 25190613 Ki = 0.9 nM T52921 CB1G6M 25190614 Ki = 0.9 nM T52921 CJLH27 25190615 Ki = 1 nM T52921 COE65V 25190616 Ki = 0.9 nM T52921 C30VGA 25190617 Ki = 1.5 nM T52921 CO7IV2 25190618 Ki = 0.8 nM T52921 C8Q7WV 25190619 Ki = 0.5 nM T52921 C0G4RJ 25190620 Ki = 6.7 nM T52921 C7X4IV 25190621 Ki = 1.4 nM T52921 CXG8O3 25190622 Ki = 0.5 nM T52921 CD5F6A 25190623 Ki = 0.4 nM T52921 CFUD47 25190624 Ki = 1.3 nM T52921 C15LIW 25190625 Ki = 0.7 nM T52921 C3LEW8 25190626 Ki = 3.6 nM T52921 CIDV61 25190627 Ki = 15.9 nM T52921 CAGS39 25190628 Ki = 1.8 nM T52921 CDS2E6 25190629 Ki = 0.6 nM T52921 CPW19O 25190630 Ki = 12.2 nM T52921 C0SBV7 25207946 Ki = 0.63 nM T52921 C21OJF 25207948 Ki = 0.3 nM T52921 C0P6CS 25207950 Ki = 0.18 nM T52921 CN9I8E 25208095 Ki = 0.2 nM T52921 C5OA1N 25208097 EC50 = 0.02512 nM T52921 C59IKP 25208099 Ki = 0.24 nM T52921 CUNA84 25208101 Ki = 0.15 nM T52921 C2WIG0 25208245 Ki = 0.22 nM T52921 CE4BI6 25208247 Ki = 1.7 nM T52921 CKNE16 25208249 Ki = 0.53 nM T52921 CB04CU 25235412 Ki = 20 nM T52921 CL2Z7J 42629117 EC50 = 14 nM T52921 CWJ2E3 43406622 IC50 > 1000 nM T52921 C49YRK 44143406 IC50 = 350 nM T52921 C3YMQ1 44143407 IC50 = 150 nM T52921 CBFR50 44143408 IC50 = 150 nM T52921 C4BOI0 44143409 IC50 = 75 nM T52921 CRL9K5 44143410 IC50 > 1000 nM T52921 CB4O2Y 44143411 IC50 > 1000 nM T52921 C0JS3Q 44143412 IC50 = 560 nM T52921 C6U7HP 44143413 IC50 = 28 nM T52921 C1TSC2 44143414 IC50 = 530 nM T52921 CAB3T9 44143415 IC50 = 37 nM T52921 CD26LJ 44143416 IC50 > 1000 nM T52921 CG3PW7 44143417 IC50 = 61 nM T52921 CB94OV 44143418 IC50 = 11 nM T52921 COP5W8 44143419 IC50 = 4 nM T52921 CY26BG 44143420 IC50 = 67 nM T52921 C8WLP6 44143421 IC50 = 270 nM T52921 C3S1PL 44143422 IC50 = 13 nM T52921 C05AWH 44143423 IC50 = 33 nM T52921 C4D0YQ 44143424 IC50 = 36 nM T52921 C5CR3I 44143425 IC50 = 72 nM T52921 CQE5U4 44143426 IC50 = 8.2 nM T52921 CZR49E 44143427 IC50 = 7.1 nM T52921 C63RXB 44143428 IC50 = 2.5 nM T52921 C8OH4S 44143429 IC50 = 4.5 nM T52921 CTE6S1 44143430 IC50 = 1.2 nM T52921 CL57VS 44143431 IC50 = 0.52 nM T52921 C2C5QW 44143432 IC50 = 0.72 nM T52921 C6GDL8 44143433 IC50 = 0.81 nM T52921 C3BNV0 44143434 IC50 = 5.7 nM T52921 CXV0B8 44143435 IC50 = 2 nM T52921 CN7HE0 44143436 IC50 = 38 nM T52921 C9CJN0 44143437 IC50 = 0.8 nM T52921 C6INT4 44143438 IC50 = 2.9 nM T52921 CJ46YA 44143439 IC50 = 23 nM T52921 CZ15CE 44143440 IC50 = 630 nM T52921 C0KB7Y 44143441 IC50 = 61 nM T52921 C3RF4I 44143442 IC50 = 27 nM T52921 CE20LQ 44143444 IC50 = 22 nM T52921 CFH9T2 44143445 IC50 = 21 nM T52921 C5NZM3 44143446 IC50 = 1.1 nM T52921 CGSW03 44143448 IC50 = 1.1 nM T52921 CBWD06 44143449 IC50 = 2.1 nM T52921 C2ST5N 44143450 IC50 = 1.4 nM T52921 CF4V5K 44143451 IC50 = 1 nM T52921 CL3R6D 44143452 IC50 = 4 nM T52921 C8IG1V 44143453 IC50 = 0.9 nM T52921 C2Q3DE 44143454 IC50 = 3.7 nM T52921 CZX75A 44143455 IC50 = 0.91 nM T52921 C02YJQ 44143456 IC50 = 1.1 nM T52921 CZV0C7 44143457 IC50 = 1.8 nM T52921 CPQ25W 44181744 Ki = 5 nM T52921 C2XE7Y 44189733 IC50 = 2.3 nM T52921 CGA8R1 44189735 IC50 = 1.9 nM T52921 C50FOG 44189834 IC50 = 2.3 nM T52921 CC63QX 44247589 Ki = 7 nM T52921 CP8Q5B 44248550 Ki = 7 nM T52921 CZNM65 44248674 Ki = 1 nM T52921 CIJF67 44248788 Ki = 272 nM T52921 C9G8KT 44248789 Ki = 34 nM T52921 C9JBR1 44248790 Ki = 22 nM T52921 C5YV0D 44248791 Ki = 14 nM T52921 C1CZ3M 44248792 Ki = 24 nM T52921 CDG15Z 44248915 Ki = 23 nM T52921 C5I7YZ 44248916 Ki = 29 nM T52921 C5T9AP 44248917 Ki = 467 nM T52921 CAY83B 44248918 Ki = 18 nM T52921 CL61MJ 44248919 Ki = 25 nM T52921 C2FLP9 44248920 Ki = 10 nM T52921 C6Q5ZF 44249045 Ki = 9 nM T52921 C0HWG8 44249046 Ki = 9 nM T52921 CHLS96 44249047 Ki = 5 nM T52921 CO4EA3 44249048 Ki = 69 nM T52921 CW6P4Y 44276782 Ki = 89 nM T52921 C9AF6B 44297435 Ki = 28.7 nM T52921 CNP5W1 44297519 Ki = 786 nM T52921 C52MGY 44297539 Ki = 0.49 nM T52921 C9UY4E 44297697 Ki = 535 nM T52921 C8F1ST 44297727 Ki = 189 nM T52921 C7ZYM4 44299404 Ki > 10000 nM T52921 CK6IY4 44315305 Ki = 10 nM T52921 CQ0OK5 44327446 EC50 = 0.7586 nM T52921 CAS38O 44332117 Ki = 4.67 nM T52921 CGZ9N2 44336905 Ki = 191 nM T52921 CYMH75 44337108 Ki = 420 nM T52921 CJ0I6Q 44337123 Ki = 64 nM T52921 CPOX86 44337129 Ki = 7222 nM T52921 CT78UG 44337131 Ki = 14 nM T52921 CO8Y5G 44337163 Ki = 745 nM T52921 CBJ01F 44337212 Ki = 49 nM T52921 C8IJM5 44337229 Ki = 26 nM T52921 C97YKG 44337230 Ki = 1062 nM T52921 C3B4WO 44337231 Ki = 1135 nM T52921 CU8IY3 44337232 Ki = 2532 nM T52921 C3M0QX 44337249 Ki = 680 nM T52921 C0MJL2 44337252 Ki = 1345 nM T52921 CB85KA 44337351 Ki = 94 nM T52921 CI13YG 44337357 Ki = 152 nM T52921 CW2FZ7 44337362 Ki = 198 nM T52921 CJ08FM 44337379 Ki = 30 nM T52921 CIP87K 44337437 Ki = 185 nM T52921 CR62KO 44337452 Ki = 79 nM T52921 C9CIP3 44337459 Ki = 3221 nM T52921 CFA2Q7 44337460 Ki = 684 nM T52921 CZP4K1 44337461 Ki = 2593 nM T52921 CF96JK 44337473 Ki = 367 nM T52921 CX87AS 44337513 Ki = 772 nM T52921 CP1VN3 44337550 Ki = 1016 nM T52921 CZ02BO 44337551 Ki = 34 nM T52921 CS9Z1O 44339374 Ki = 225 nM T52921 C73CSH 44339393 Ki = 153 nM T52921 CF08RA 44339398 Ki > 10000 nM T52921 CFNR91 44339423 Ki = 33 nM T52921 CW56BK 44339424 Ki = 12 nM T52921 C4POK5 44339425 Ki = 135 nM T52921 C03PDA 44339449 Ki = 692 nM T52921 CGI10R 44339450 Ki = 715 nM T52921 C7HIP9 44339463 Ki = 879 nM T52921 CQ24IT 44339491 Ki > 10000 nM T52921 CC1VG7 44339500 Ki = 234 nM T52921 C73QPW 44339504 Ki = 502 nM T52921 CABQ05 44339505 Ki = 1270 nM T52921 C7GRF4 44339525 Ki = 1194 nM T52921 CY85GQ 44339526 Ki = 6520 nM T52921 CZRJ83 44339528 Ki > 10000 nM T52921 CKP7R5 44339529 Ki > 10000 nM T52921 CAD1O4 44339530 Ki = 1106 nM T52921 CIZU20 44339531 Ki > 10000 nM T52921 C2LQO7 44339540 Ki = 307 nM T52921 C7E4MS 44339576 Ki = 47 nM T52921 C2PDT6 44339596 Ki = 102 nM T52921 C34DEN 44339684 Ki = 82 nM T52921 CO3C7M 44339695 Ki = 12 nM T52921 CGY16P 44339707 Ki = 827 nM T52921 CD9ZS8 44342270 IC50 = 1910 nM T52921 C4BK0O 44352743 EC50 = 439 nM T52921 CHX36W 44352744 EC50 = 286 nM T52921 C9RN1Y 44352745 IC50 = 2710 nM T52921 C1GZ8E 44352920 IC50 = 874 nM T52921 CD18TR 44366689 Ki = 2130 nM T52921 CYL95J 44366690 Ki = 35 nM T52921 C7IFR8 44366822 Ki = 34 nM T52921 CL1JV2 44366823 Ki = 44 nM T52921 CX7A3N 44388460 EC50 = 0.06607 nM T52921 CLV18K 44388461 EC50 = 0.1 nM T52921 CK95WL 44388462 EC50 = 0.06761 nM T52921 C5FA4H 44388465 EC50 = 0.4786 nM T52921 CBUS05 44388466 EC50 = 0.2399 nM T52921 CJG21X 44388467 EC50 = 0.2089 nM T52921 CZ7L6C 44388472 EC50 = 5.888 nM T52921 C4WRI8 44388474 EC50 = 0.4074 nM T52921 C5I7AN 44390989 Ki = 12 nM T52921 C2TP3J 44390999 Ki = 620 nM T52921 C9FBO3 44391012 Ki = 1115 nM T52921 C2W7BJ 44391023 Ki = 282 nM T52921 C4BF2U 44391031 Ki = 905 nM T52921 CF49QH 44391052 Ki = 32 nM T52921 C7A8DM 44391062 Ki = 10.8 nM T52921 CTA04B 44391063 Ki = 462 nM T52921 C1WGX6 44391067 Ki = 52 nM T52921 C8Y7OV 44391069 Ki = 218 nM T52921 CT8W3P 44391075 Ki = 1920 nM T52921 CY7OH0 44391079 Ki = 42 nM T52921 CPZ7L8 44391081 Ki = 28 nM T52921 CR5TN7 44391092 Ki = 37 nM T52921 C2DB4N 44391093 Ki = 768 nM T52921 CO2T5M 44391094 Ki = 14 nM T52921 CL79EO 44391099 Ki = 838 nM T52921 C3HTZ1 44391102 Ki = 509 nM T52921 CW76ZY 44391103 Ki = 24 nM T52921 CN1LD9 44391104 Ki = 38.2 nM T52921 CD3QV8 44391111 Ki = 60 nM T52921 CK2HV1 44391119 Ki = 113 nM T52921 C8RDV5 44391124 Ki = 3 nM T52921 C1UDL9 44391133 Ki = 20 nM T52921 CSV6X2 44391134 Ki = 25 nM T52921 CJ9MX1 44391137 Ki = 815 nM T52921 C18SDI 44391138 Ki = 126 nM T52921 C6ZF9E 44391155 Ki = 8.3 nM T52921 CY6T4F 44391156 Ki = 108 nM T52921 CJB0U8 44391157 Ki = 39 nM T52921 C5ZFX2 44394283 Ki = 231 nM T52921 COB70L 44394284 Ki = 40 nM T52921 C5BTZ1 44394320 Ki = 1878 nM T52921 C6DB4X 44394324 Ki = 28.7 nM T52921 C2OV9B 44394344 Ki = 46 nM T52921 C1Y3NV 44394345 Ki = 2614 nM T52921 CCR2U1 44394375 Ki = 83 nM T52921 CQ2O6J 44394381 Ki = 3.9 nM T52921 CTJ2I9 44394405 Ki = 63 nM T52921 CLFU54 44394419 Ki = 187 nM T52921 C0A1OW 44394487 Ki = 5 nM T52921 C61AXY 44394529 Ki = 9535 nM T52921 CRCV49 44394559 Ki = 609 nM T52921 C3YD8C 44395259 Ki > 10000 nM T52921 CR8AF5 44395265 Ki > 10000 nM T52921 CI7GR3 44395286 Ki = 149 nM T52921 CLB5E3 44395291 Ki > 10000 nM T52921 CEX0W2 44395306 Ki = 590 nM T52921 C69ACH 44395319 Ki > 10000 nM T52921 CQO0Y5 44395366 Ki > 10000 nM T52921 C0FUP2 44395387 Ki > 10000 nM T52921 C06LKH 44395410 Ki = 372 nM T52921 C7GP1E 44404646 IC50 = 290 nM T52921 CILB28 44404652 IC50 = 380 nM T52921 C38GAM 44404653 IC50 = 1310 nM T52921 CA58SU 44404670 IC50 = 120 nM T52921 C83PCH 44404679 IC50 = 100 nM T52921 CU0YX9 44404684 IC50 = 2400 nM T52921 CEJ7F8 44404689 IC50 = 2680 nM T52921 CD8M2R 44404693 IC50 = 710 nM T52921 C5X8YK 44404694 IC50 = 470 nM T52921 CODG94 44404695 IC50 = 150 nM T52921 CD79WM 44404698 IC50 = 450 nM T52921 C0BED6 44404699 IC50 = 37 nM T52921 CGA15Y 44404706 IC50 = 10000 nM T52921 C2NHS0 44404707 IC50 > 10000 nM T52921 CJCY60 44404711 IC50 = 1080 nM T52921 CK73OG 44404721 IC50 = 350 nM T52921 CNX5T8 44404731 IC50 = 180 nM T52921 CW9QG2 44406457 IC50 > 10000 nM T52921 CGN73V 44406458 IC50 > 10000 nM T52921 C0J7IK 44406489 IC50 = 6000 nM T52921 C5TIM4 44406497 IC50 = 1000 nM T52921 CBUR32 44406503 IC50 = 10000 nM T52921 C17FYG 44406538 IC50 = 15000 nM T52921 C07CNE 44406539 IC50 = 7000 nM T52921 C5DGV2 44406540 IC50 = 3850 nM T52921 C9Z0ET 44406541 IC50 > 10000 nM T52921 C1L8CG 44406543 IC50 = 10400 nM T52921 CP1OZ6 44406544 IC50 > 10000 nM T52921 CS04TK 44406550 IC50 = 5800 nM T52921 C8HRC9 44406551 IC50 = 15000 nM T52921 CSPE30 44406557 IC50 = 13400 nM T52921 CD7Y0Z 44406585 IC50 > 10000 nM T52921 CC15BY 44406587 IC50 = 10000 nM T52921 C1IM9R 44406603 IC50 = 1000 nM T52921 C3VE8N 44406604 IC50 = 1000 nM T52921 CCI5Z1 44406618 IC50 = 300 nM T52921 C7ES2W 44406621 IC50 = 130 nM T52921 C0SKT9 44406641 IC50 > 10000 nM T52921 C38ABN 44406682 IC50 > 10000 nM T52921 CZ65PF 44406685 IC50 > 10000 nM T52921 CWY76P 44406719 IC50 = 4000 nM T52921 CP5H7S 44406907 IC50 > 1000 nM T52921 CHKO45 44406969 IC50 > 1000 nM T52921 CV4C6R 44406970 IC50 > 1000 nM T52921 C7BNY9 44406975 IC50 > 1000 nM T52921 C0W1EN 44406978 IC50 > 1000 nM T52921 C5U7KF 44406979 IC50 > 1000 nM T52921 CM31XO 44406989 IC50 > 1000 nM T52921 CC0H4U 44406991 IC50 > 1000 nM T52921 CNP5V6 44406994 IC50 > 1000 nM T52921 C3BQ7S 44406995 IC50 > 1000 nM T52921 C92ZTH 44406996 IC50 > 1000 nM T52921 CN82CH 44406997 IC50 > 1000 nM T52921 CX20ZA 44406998 IC50 > 1000 nM T52921 CMRF31 44407013 IC50 = 630 nM T52921 C8RNE9 44407016 IC50 > 1000 nM T52921 CA2OD1 44407020 IC50 = 870 nM T52921 C0OB8F 44407023 IC50 > 1000 nM T52921 C21UFE 44407028 IC50 > 1000 nM T52921 C8GK1Q 44407036 IC50 > 1000 nM T52921 CGO7M0 44407037 IC50 > 1000 nM T52921 C4YW1C 44407038 IC50 > 1000 nM T52921 C4QT3D 44407040 IC50 > 1000 nM T52921 CK84HW 44407043 IC50 > 1000 nM T52921 CZ8D9R 44407044 IC50 = 30 nM T52921 C7QWZ5 44407048 IC50 = 360 nM T52921 CYJ04D 44407049 IC50 > 1000 nM T52921 CJ4A2W 44407050 IC50 > 1000 nM T52921 CU20IA 44407063 IC50 > 1000 nM T52921 C5PDG8 44407065 IC50 > 1000 nM T52921 CGAD30 44407066 IC50 > 1000 nM T52921 CT49JG 44407070 IC50 = 170 nM T52921 C9WJZ5 44407074 IC50 > 1000 nM T52921 CW2CP3 44407078 IC50 > 1000 nM T52921 CL9QK6 44407080 IC50 > 1000 nM T52921 C2S5NT 44407081 IC50 > 1000 nM T52921 C0QB6E 44407084 IC50 = 131 nM T52921 CLG4Y9 44407085 IC50 = 230 nM T52921 CPQ7H2 44407086 IC50 = 290 nM T52921 C0K7ZH 44407091 IC50 > 1000 nM T52921 CM8JK6 44407109 IC50 > 1000 nM T52921 C8R1QN 44407112 IC50 = 340 nM T52921 CEZ4I2 44407113 IC50 > 1000 nM T52921 CA3OW4 44407116 IC50 = 21 nM T52921 CLE6W9 44407119 IC50 > 1000 nM T52921 CK4NE2 44407129 IC50 = 50 nM T52921 CKUT49 44407133 IC50 = 24 nM T52921 COS85F 44407140 IC50 = 330 nM T52921 CAMX28 44407145 IC50 > 1000 nM T52921 CRP3D2 44407146 IC50 > 1000 nM T52921 CZO5R6 44407156 IC50 = 900 nM T52921 C2YME3 44413175 IC50 > 1000 nM T52921 CM7LE4 44413183 IC50 > 1000 nM T52921 C0M9TX 44413184 IC50 > 1000 nM T52921 CFJ64A 44413232 Ki = 970 nM T52921 CNFC81 44413248 Ki > 5000 nM T52921 C0V4FI 44413286 Ki = 550 nM T52921 CS7BI8 44413301 Ki = 81 nM T52921 C1NGS0 44413314 Ki = 94 nM T52921 C5J0BU 44413315 Ki > 5000 nM T52921 CH7E1C 44413329 Ki > 5000 nM T52921 C1OQ0L 44413330 Ki = 2 nM T52921 CKV5S0 44413361 Ki = 52 nM T52921 C5PHK7 44413362 Ki = 62 nM T52921 CSQZ28 44413379 Ki > 5000 nM T52921 CCU2B5 44413384 Ki = 660 nM T52921 CD5SZ9 44413385 Ki = 57 nM T52921 C7GE2K 44413395 Ki > 5000 nM T52921 CCK6Y5 44413396 Ki = 1650 nM T52921 C0FL8K 44413401 Ki = 3500 nM T52921 C6J3HP 44413402 Ki > 5000 nM T52921 CB2OJ9 44413408 Ki = 160 nM T52921 C82VJB 44413413 Ki > 5000 nM T52921 CP31JV 44413414 Ki = 820 nM T52921 C98OQG 44413423 Ki > 5000 nM T52921 CH0DS7 44413441 Ki = 710 nM T52921 CLSK72 44413442 Ki = 10 nM T52921 C6O2VL 44414730 IC50 > 10000 nM T52921 C5Z9VE 44414845 IC50 > 10000 nM T52921 C4LI9Q 44414865 IC50 > 10000 nM T52921 C10OMS 44426811 Ki = 9 nM T52921 C49KAS 44426813 Ki = 41 nM T52921 CJK6Y5 44426815 Ki = 4035 nM T52921 CJ5FC0 44426816 Ki = 295 nM T52921 C4TFP1 44426818 Ki = 1887 nM T52921 CP1Z5J 44426819 Ki = 10000 nM T52921 CP5V8D 44426821 Ki = 8183 nM T52921 C5L4SE 44426822 Ki = 214 nM T52921 C36SCP 44426823 Ki = 323 nM T52921 C72RXV 44426824 Ki = 35 nM T52921 C0S5TE 44426829 Ki = 12 nM T52921 CL1EG2 44426830 Ki = 357 nM T52921 CBFY73 44426831 Ki = 225 nM T52921 CFO9Q6 44426832 Ki = 0.6 nM T52921 C2NFA4 44426833 Ki = 26 nM T52921 COJ48Z 44426834 Ki = 132 nM T52921 CUD42S 44426835 Ki = 5 nM T52921 CKJ90O 44426836 Ki = 11 nM T52921 CZ4R6J 44426837 Ki = 125 nM T52921 CPDE73 44426838 Ki = 9 nM T52921 C53JGK 44426839 Ki = 6753 nM T52921 C7IJY0 44426840 Ki = 6 nM T52921 CJB90W 44426841 Ki = 42 nM T52921 C4Z1FX 44426842 Ki = 21 nM T52921 CK3B6E 44426843 Ki = 3 nM T52921 CD3TB8 44426844 Ki = 439 nM T52921 CF5OJ0 44430021 Ki = 1449 nM T52921 CUQ95Y 44430022 Ki = 16 nM T52921 CZA0E6 44430023 Ki = 1.6 nM T52921 CWX67P 44430033 Ki = 15 nM T52921 C40BHT 44430038 Ki = 0.4 nM T52921 C1QXR6 44430040 Ki = 0.7 nM T52921 CS6Y5Z 44430042 Ki = 0.5 nM T52921 C4CHV5 44430043 Ki = 1.1 nM T52921 CX9P5R 44430044 Ki = 0.5 nM T52921 CA51JN 44430045 Ki = 110 nM T52921 C2G9HQ 44430046 Ki = 674 nM T52921 C8PI4A 44430047 Ki = 9.6 nM T52921 CL1N4D 44430048 Ki = 4.6 nM T52921 C0AYM6 44430049 Ki = 5.5 nM T52921 CMJT74 44430050 Ki = 0.7 nM T52921 C4ZG6A 44430079 Ki = 2 nM T52921 CSNQ43 44430080 Ki = 12 nM T52921 CXV9J7 44430081 Ki = 5.9 nM T52921 CFHY18 44430083 Ki = 1.9 nM T52921 C6SBE1 44430084 Ki = 2.2 nM T52921 CXZ2D3 44430085 Ki = 0.9 nM T52921 CI4X3Z 44430087 Ki = 0.6 nM T52921 C8D0ZX 44431782 Ki = 1273 nM T52921 CT30KJ 44437601 Ki = 3 nM T52921 C1EHS4 44437602 Ki = 2 nM T52921 CX5O0J 44437604 Ki = 5 nM T52921 CWOJ02 44437605 Ki = 3 nM T52921 CK73VO 44437606 Ki = 3 nM T52921 CJ1ST3 44437610 Ki = 0.5 nM T52921 CFH6A5 44437613 Ki = 22 nM T52921 C0M9SC 44437615 Ki = 4 nM T52921 CFN8Z9 44437617 Ki = 6 nM T52921 CTK2S0 44437619 Ki = 1 nM T52921 C4PK1O 44437623 Ki = 5 nM T52921 CP4HR6 44437626 Ki = 4 nM T52921 CA5S2P 44437627 Ki = 46 nM T52921 CKEG06 44437628 Ki = 12 nM T52921 CT7V0O 44437629 Ki = 1595 nM T52921 C45ZTN 44437630 Ki = 10 nM T52921 CQKL94 44437636 Ki = 4 nM T52921 C43URV 44437637 Ki = 3 nM T52921 CJ8L4A 44437638 Ki = 2 nM T52921 CNBQ93 44437639 Ki = 5 nM T52921 C2AV5I 44437640 Ki = 19 nM T52921 CN3R5G 44437641 Ki = 29 nM T52921 C6NA9R 44437642 Ki = 20 nM T52921 CH5RW4 44437643 Ki = 155 nM T52921 C7RIC8 44437644 Ki = 15 nM T52921 C5IL8O 44437645 Ki = 20 nM T52921 CX1S4V 44437646 Ki = 12 nM T52921 CV19NL 44437647 Ki = 29 nM T52921 C02YET 44437648 Ki = 12 nM T52921 CJ2PH5 44437649 Ki = 3 nM T52921 CVH1I9 44437652 Ki = 23 nM T52921 C0ME9B 44437654 Ki = 2 nM T52921 CRKH10 44437656 Ki = 2 nM T52921 CZB4Q9 44438912 Ki = 61.2 nM T52921 CP85QV 44438914 Ki = 824 nM T52921 C7RD2E 44438916 Ki = 14 nM T52921 CNL30S 44438917 Ki = 3.2 nM T52921 C5D4NZ 44438920 Ki = 3.5 nM T52921 CA2LD5 44438921 Ki = 17 nM T52921 C6H7AD 44438922 Ki = 2.4 nM T52921 CRN3W4 44438961 Ki = 1.1 nM T52921 CGYD89 44438962 Ki = 1.5 nM T52921 CZ48KD 44438963 Ki = 36.5 nM T52921 C2EGK7 44438964 Ki = 10.8 nM T52921 COX57F 44438965 Ki = 9 nM T52921 C9S2HB 44438966 Ki = 11.5 nM T52921 C1HF6E 44438967 Ki = 140 nM T52921 C3L7SB 44438968 Ki = 9 nM T52921 CE63GK 44438971 Ki = 249 nM T52921 C8TVI4 44438974 Ki = 6.3 nM T52921 CPHS56 44438975 Ki = 250 nM T52921 CK3Z5G 44438978 Ki = 49 nM T52921 CPA4U5 44438983 Ki = 0.3 nM T52921 C2TKY5 44438988 Ki = 0.8 nM T52921 CL7WN5 44438993 Ki = 2.6 nM T52921 C0A2OM 44439000 Ki = 1.4 nM T52921 CMQA60 44439001 Ki = 8.4 nM T52921 CN4KX9 44449764 IC50 = 31 nM T52921 CWN0C3 44449766 IC50 = 78 nM T52921 CE97XC 44449767 IC50 = 180 nM T52921 C7NKJ3 44449771 IC50 = 140 nM T52921 CRO1B7 44449793 IC50 = 2900 nM T52921 CTMI71 44449822 IC50 = 63 nM T52921 CU6I5Y 44449823 IC50 > 10000 nM T52921 C8QE6N 44449850 IC50 = 8200 nM T52921 CH5MN1 44449851 IC50 = 910 nM T52921 CT39QP 44450085 IC50 = 1.8 nM T52921 C1SQ7M 44450086 IC50 = 20 nM T52921 CGN7O0 44450151 IC50 = 15 nM T52921 CS4DO9 44450180 IC50 = 240 nM T52921 CL5K3J 44450207 IC50 = 2900 nM T52921 CK41RX 44450208 IC50 = 140 nM T52921 CUR83O 44450209 IC50 = 380 nM T52921 C37FVM 44450210 IC50 = 55 nM T52921 CL78ZG 44451517 Ki = 3.548 nM T52921 CG2WD7 44451518 Ki = 21.88 nM T52921 CBK6R5 44451542 Ki = 3.89 nM T52921 CC36BM 44451543 Ki = 2.512 nM T52921 CKB0F9 44451569 Ki = 1.698 nM T52921 C2EJP0 44451572 Ki = 28.84 nM T52921 CYQ53B 44451573 Ki = 1174.9 nM T52921 CGJ3R8 44451592 Ki = 7.943 nM T52921 CAC1G4 44451593 Ki = 17.38 nM T52921 CV26FM 44451594 Ki = 4.898 nM T52921 CKRM60 44451595 Ki = 1.514 nM T52921 C4S0BF 44451619 Ki = 2.399 nM T52921 CAVN40 44451620 Ki = 912.01 nM T52921 C2NCL3 44451621 Ki = 1.202 nM T52921 CHPO59 44451647 Ki = 95.5 nM T52921 C70TSK 44451648 Ki = 11.75 nM T52921 CZ1R2D 44451649 Ki = 0.8913 nM T52921 C5UM1O 44451650 Ki = 1.995 nM T52921 CF4SX9 44451673 Ki = 37.15 nM T52921 C3O8ZP 44451696 Ki = 29.51 nM T52921 C7VLH3 44451724 Ki = 41.69 nM T52921 CYIP73 44451748 Ki = 1.862 nM T52921 C2IS4W 44451777 Ki = 4.898 nM T52921 CST06H 44451779 Ki = 3.311 nM T52921 C4C9TD 44451805 Ki = 4.169 nM T52921 C5RLP6 44451837 Ki = 3.715 nM T52921 CO01GQ 44451872 Ki = 5.888 nM T52921 C7KL9C 44451895 Ki = 9.55 nM T52921 C25JHV 44451918 Ki = 1.413 nM T52921 C4DL5C 44469677 IC50 > 10000 nM T52921 CFAZ41 44517710 IC50 = 5.6 nM T52921 C6T1UX 44551464 EC50 = 3.6 nM T52921 CC01KM 44561020 Ki = 3.7 nM T52921 CY14MD 44561518 Ki = 6 nM T52921 CPO2R3 44570675 Ki = 2.5 nM T52921 CNUJ50 44574003 IC50 = 38 nM T52921 C1T4QN 44574053 IC50 = 16 nM T52921 CW8DR7 44574393 Ki = 1571 nM T52921 C67IZG 44574538 Ki = 3 nM T52921 C5Q4HZ 44574539 Ki = 7.3 nM T52921 C74LHO 44574585 Ki = 2.7 nM T52921 CPL5V1 44574586 Ki = 5.2 nM T52921 C7K4PC 44574587 Ki = 13 nM T52921 C1JPH8 44574588 Ki = 1.9 nM T52921 CNCS12 44574629 Ki = 3.6 nM T52921 CJXE09 44574630 Ki = 14 nM T52921 C2FO5H 44574631 Ki = 3 nM T52921 C5YQ6B 44574632 Ki = 7.4 nM T52921 CD18EP 44574671 Ki = 385 nM T52921 CDS1G8 44574672 Ki = 8 nM T52921 C6ZMS9 44574705 Ki = 6 nM T52921 CDNP82 44574706 Ki = 3151 nM T52921 C13RZI 44574707 Ki = 100 nM T52921 CXQM01 44574708 Ki = 3 nM T52921 CW1GU7 44574743 Ki = 6 nM T52921 CL6UI1 44574744 Ki = 4 nM T52921 CKO8N4 44574745 Ki = 2 nM T52921 CLVU91 44574789 Ki = 11 nM T52921 C5JZK9 44574790 Ki = 5.3 nM T52921 CVZ6K3 44574848 Ki = 31 nM T52921 C1MWD8 44574849 Ki = 40 nM T52921 CA78KV 44574850 Ki = 22 nM T52921 CX1BL6 44574851 Ki = 285 nM T52921 C7YAD5 44574889 Ki = 678 nM T52921 CPH7D4 44574890 Ki = 4.9 nM T52921 CQL2E4 44574891 Ki = 7 nM T52921 C9C3ZJ 44574892 Ki = 10 nM T52921 CLG57R 44574958 Ki = 12 nM T52921 CLMH36 44574962 Ki = 8.2 nM T52921 CAW3R4 44574963 Ki = 11 nM T52921 CAWB12 44575043 Ki = 17 nM T52921 CZO5J4 44575091 Ki = 908 nM T52921 CI6Y7U 44575092 Ki = 142 nM T52921 CO26ZW 44576625 IC50 = 8 nM T52921 CSH8K2 44576626 IC50 = 59 nM T52921 CD0T5K 44576627 IC50 = 18 nM T52921 C4ZCX6 44576628 IC50 = 1.1 nM T52921 CR0LN1 44593575 Ki = 198 nM T52921 CTYR04 44593576 Ki = 19 nM T52921 CDPU87 44596170 EC50 = 94 nM T52921 C45PUQ 45102745 Ki = 0.7 nM T52921 CU8I6T 45263517 Ki = 0.7 nM T52921 CVDQ53 45265789 Ki = 23 nM T52921 C6VZM4 45267505 IC50 = 2.5 nM T52921 CA2MH1 45267506 IC50 = 33 nM T52921 CK16EZ 45267601 IC50 = 28 nM T52921 CR59UW 45267616 IC50 = 200 nM T52921 CY4UA3 45267639 IC50 > 1000 nM T52921 CA2O3N 45268153 Ki = 3 nM T52921 C4F6IO 45268355 IC50 = 4.3 nM T52921 CX3YO5 45268356 IC50 = 17 nM T52921 C7UG6Q 45268498 IC50 = 2.3 nM T52921 C8QG3U 45268503 IC50 = 160 nM T52921 C3YEJ9 45268504 IC50 = 33 nM T52921 C8BPX4 45269032 Ki = 2 nM T52921 CKC09D 45269228 IC50 = 210 nM T52921 CKZ35F 45269347 IC50 > 1000 nM T52921 C06ITN 45269349 IC50 > 1000 nM T52921 C78UOX 45269357 IC50 = 4.7 nM T52921 C4WT5J 45269358 IC50 = 1.4 nM T52921 C3I6YO 45269372 IC50 = 160 nM T52921 CSL62Z 45270082 IC50 = 6.4 nM T52921 C6PRX0 45270174 IC50 = 620 nM T52921 C6GRC1 45270175 IC50 > 1000 nM T52921 CA38NB 45270184 IC50 = 3.7 nM T52921 CVU53F 45270190 IC50 > 1000 nM T52921 CA3S7Q 45270196 IC50 = 530 nM T52921 CY79OE 45270202 IC50 = 540 nM T52921 CVP80J 45270203 IC50 = 500 nM T52921 CC5I8O 45270712 Ki = 71 nM T52921 CM5ZI0 45270907 IC50 = 2 nM T52921 C6P0AZ 45270917 IC50 = 13 nM T52921 CDT5G6 45270928 IC50 = 15 nM T52921 C8KS5V 45271014 IC50 = 850 nM T52921 C2G5XK 45271015 IC50 = 26 nM T52921 CO05CL 45271041 IC50 = 11 nM T52921 CU84PI 45271534 Ki = 2 nM T52921 CP6V4Q 45271862 IC50 = 520 nM T52921 CMGB49 45271885 IC50 = 190 nM T52921 CJGX41 45271896 IC50 > 1000 nM T52921 C6G9DQ 45271902 IC50 = 160 nM T52921 C1UOZ9 45272626 IC50 = 7.8 nM T52921 C0P6GI 45272729 IC50 > 1000 nM T52921 CL0Y5P 45272733 IC50 > 1000 nM T52921 C09HIZ 45272755 IC50 > 1000 nM T52921 CFU9R4 45273531 IC50 = 0.61 nM T52921 CX0N4V 45273537 IC50 = 3.1 nM T52921 CJNO02 45273546 IC50 = 1.4 nM T52921 C3ZPJ5 45273547 IC50 = 12 nM T52921 CGT48R 45273662 IC50 = 130 nM T52921 C91JXR 45273672 IC50 > 1000 nM T52921 C58HQB 45273679 IC50 = 4.5 nM T52921 CS0GA2 45273702 IC50 = 96 nM T52921 C3YHF0 46227961 EC50 = 135 nM T52921 C7LW1S 46227963 Ki = 4.2 nM T52921 C9L6WI 46227966 EC50 = 15 nM T52921 CA2P9C 46879475 Ki = 4082 nM T52921 CH45JY 46879476 Ki = 454 nM T52921 CS2V6N 46879477 Ki = 16 nM T52921 C6R8JO 46879478 Ki = 106 nM T52921 C9URN3 46879536 Ki = 21 nM T52921 C5PW9I 46879537 Ki = 11 nM T52921 CW2N7P 46879538 Ki = 2.9 nM T52921 CGJS91 46879539 Ki = 6.4 nM T52921 C08CHW 46879578 Ki = 28 nM T52921 CNF9D6 46879579 Ki = 2.3 nM T52921 C8UD2Z 46879580 Ki = 0.6 nM T52921 C9E8YP 46879581 Ki = 2.5 nM T52921 C9GB7O 46879627 Ki = 2152 nM T52921 C5VKU0 46879628 Ki = 227 nM T52921 CU2F0K 46879629 Ki = 111 nM T52921 CS7BP4 46879630 Ki = 295 nM T52921 C06NBW 46879667 Ki = 44 nM T52921 C0WY3K 46879668 Ki = 22 nM T52921 C5L7DB 46879669 Ki = 7.7 nM T52921 CSG31K 46879670 Ki = 5 nM T52921 C7P4UE 46879716 Ki = 7.1 nM T52921 CQSI16 46879992 Ki = 470 nM T52921 C16INW 46879993 Ki = 227 nM T52921 C9NR8Q 46880030 Ki = 35 nM T52921 C0O1PU 46880031 Ki = 15 nM T52921 CDY2L8 46880032 Ki = 0.2 nM T52921 CK01VS 46880033 Ki = 1.3 nM T52921 CFXU43 46880088 Ki = 62 nM T52921 CDM4C0 46880089 Ki = 5.2 nM T52921 CA8JU6 46880090 Ki = 5.5 nM T52921 C7LX9B 46880114 Ki = 4.7 nM T52921 CX7RS8 46880115 Ki = 253 nM T52921 C2VS0K 46880116 Ki = 3.5 nM T52921 C18JDU 46880117 Ki = 487 nM T52921 CHN70E 46880151 Ki = 2560 nM T52921 CI5D6H 46880152 Ki = 259 nM T52921 CF0ER7 46880153 Ki = 1118 nM T52921 CU8JO5 46880154 Ki = 471 nM T52921 CR35XL 46880155 Ki = 186 nM T52921 CI6ZA1 46880237 Ki = 29 nM T52921 CID57V 46880238 Ki = 2.7 nM T52921 CG6UO7 46880239 Ki = 18 nM T52921 C31BLP 46880240 Ki = 1050 nM T52921 C3T6NH 49843555 Ki = 1.438 nM T52921 C0TCI3 52915030 IC50 = 31.6 nM T52921 CK6GN5 52915031 IC50 = 28.1 nM T52921 CXF14W 52915032 IC50 = 32.7 nM T52921 CELZ30 52915143 IC50 = 98.9 nM T52921 CR57AK 52915144 IC50 = 308.9 nM T52921 CP29EV 52915145 IC50 = 186.2 nM T52921 C15YXV 52915146 IC50 = 208.6 nM T52921 C45JNG 52915147 IC50 = 141.9 nM T52921 COM38Z 52915266 IC50 = 146.5 nM T52921 COEU73 52915267 IC50 = 154.5 nM T52921 CZK59C 52915268 IC50 = 184.5 nM T52921 C27KOF 52915269 IC50 = 83 nM T52921 CQ71YX 52915270 IC50 = 1115.9 nM T52921 CH56XF 52915389 IC50 = 731.6 nM T52921 C02UBO 52915390 IC50 = 1217.8 nM T52921 CP2M6E 52915391 IC50 = 667.5 nM T52921 CPA43I 52915392 IC50 = 482.9 nM T52921 C5OA9H 52915393 IC50 = 304.6 nM T52921 CA3P2C 52915514 IC50 = 404.7 nM T52921 CK39TQ 52915515 IC50 = 159.6 nM T52921 C98UZW 52915516 IC50 = 799.8 nM T52921 CLAS61 52915517 IC50 = 206.9 nM T52921 C7FDE9 52915518 IC50 = 1106.7 nM T52921 C9YOD2 52915634 IC50 = 246.4 nM T52921 C1ZHF3 52915635 IC50 = 144 nM T52921 CZB67C 52915636 IC50 = 211.6 nM T52921 CE3IS2 52915637 IC50 = 152.9 nM T52921 C8F0TA 52916174 IC50 = 207.3 nM T52921 C4K3NO 52916266 IC50 = 115.7 nM T52921 CPV9S3 52916267 IC50 = 48 nM T52921 CXGN56 52916358 IC50 = 35.6 nM T52921 CO4Q6E 52916359 IC50 = 50.9 nM T52921 CM0KA5 52916360 IC50 = 83.3 nM T52921 CN8L4T 52916470 IC50 = 63.1 nM T52921 C96OUY 52916471 IC50 = 113.6 nM T52921 CC92WA 52916472 IC50 = 82.7 nM T52921 CG91EA 52916597 IC50 = 82.1 nM T52921 CYB6J8 52916598 IC50 = 76.5 nM T52921 CG1F9W 52916599 IC50 = 56.6 nM T52921 C7NO2D 52916712 IC50 = 76.2 nM T52921 CZ3K9S 52916713 IC50 = 71.7 nM T52921 CI32WO 52916714 IC50 = 30.1 nM T52921 C4FZT7 52951674 Ki = 0.231 nM T52921 CS4T2C 52951675 Ki = 0.101 nM T52921 C5VLO1 52951807 Ki = 0.106 nM T52921 CK7I1T 52951808 Ki = 0.137 nM T52921 C0UVH3 52951809 Ki = 0.09 nM T52921 C40BPO 52951810 Ki = 0.15 nM T52921 CF0L7D 52951938 Ki = 4.51 nM T52921 CDAN40 52951939 Ki = 17.1 nM T52921 C89QXK 52951940 Ki = 5.61 nM T52921 COVP24 52951941 Ki = 10.2 nM T52921 CR6B4G 52951942 Ki = 9.08 nM T52921 CSF4G7 52952043 Ki = 5.32 nM T52921 CTU43X 53316968 Ki = 4.54 nM T52921 CCOD69 53316969 Ki = 4.29 nM T52921 CI6CQ0 53319615 Ki = 0.15 nM T52921 C6SY4G 53319616 Ki = 80.5 nM T52921 C3PW1V 53319617 Ki = 4.29 nM T52921 C2EV1S 53322245 Ki = 0.96 nM T52921 C1L8IV 53322246 Ki > 250 nM T52921 C0MD2H 53324890 Ki = 0.73 nM T52921 C5E7LW 53325608 Ki = 4.29 nM T52921 CRZ76L 53326167 Ki = 6.56 nM T52921 CJ46YH 54580478 Ki = 58.88 nM T52921 C35VCH 54580479 Ki = 48.98 nM T52921 CED95R 54581495 Ki = 107.15 nM T52921 CW7FV5 54581497 Ki = 83.18 nM T52921 CWOA13 54583469 Ki > 10000 nM T52921 CE9OC2 54584439 Ki = 60.26 nM T52921 CA4XQ2 54584440 Ki = 1148.15 nM T52921 C8J5OH 54585395 Ki = 58.88 nM T52921 CM3A1U 54585396 Ki = 158.49 nM T52921 CYS7J8 54586351 Ki > 10000 nM T52921 CROS84 54756989 Ki = 18.5 nM T52921 C2ISE6 54756990 Ki = 22 nM T52921 CCN2E8 56658044 Ki = 16 nM T52921 C69VIF 56661555 Ki = 67.8 nM T52921 CDKP63 56664973 Ki = 8.46 nM T52921 C4QM3N 56668405 Ki = 237 nM T52921 CX8F2N 56681954 Ki = 133 nM T52921 C2A4MQ 56681955 Ki = 159 nM T52921 CQY16A 57391870 Ki > 10000 nM T52921 CI5H3N 58268566 Ki = 0.0916 nM T52921 C6Z9JF 58268629 Ki = 0.0892 nM T52921 C6G5TY 60154189 Ki = 7.37 nM T52921 C2ZG0F 60154190 Ki = 9.4 nM T52921 C8MS6N 60154191 Ki = 1.84 nM T52921 CW63KM 60154192 Ki = 5.16 nM T52921 C2QX6R 60154193 Ki > 10 nM T52921 CTCJ21 60154194 Ki > 10 nM T52921 CO4Q8V 60154195 Ki > 10 nM T52921 C80XNK 60154196 Ki > 10 nM T52921 CJ8DW1 60154197 Ki > 40 nM T52921 CD5R7A 60154198 Ki > 40 nM T52921 CY1U7F 60154199 Ki > 40 nM T52921 CXRV52 60154200 Ki = 0.396 nM T52921 CD46EJ 60154264 Ki = 0.114 nM T52921 C98XRD 66911347 Ki = 205 nM T52921 CZ63PG 66986460 Ki = 3.7 nM T52921 CF5I0R 68917692 Ki = 1.26 nM T52921 CPE62M 70682348 Ki > 250 nM T52921 C6KD9C 70682349 Ki > 250 nM T52921 C2PC8W 70682350 Ki > 250 nM T52921 C58AOU 70682351 Ki = 9.84 nM T52921 CH42QP 70682760 Ki = 0.194 nM T52921 C6G0SO 70684433 Ki = 11.6 nM T52921 CZ5B7A 70684434 Ki > 250 nM T52921 CLY56A 70684435 Ki > 250 nM T52921 C8U1PW 70684436 Ki = 13.6 nM T52921 C4ZU7H 70684841 Ki = 0.0902 nM T52921 C6DC8G 70684842 Ki = 0.0672 nM T52921 CWAL85 70686573 Ki > 250 nM T52921 CAFB10 70686574 Ki > 250 nM T52921 CZ6E9M 70686575 Ki > 250 nM T52921 CPD35T 70686907 Ki = 5.32 nM T52921 CI61FE 70688692 Ki > 250 nM T52921 C08OUK 70688693 Ki > 250 nM T52921 CMKZ80 70688694 Ki > 250 nM T52921 CLK7P0 70688695 Ki > 250 nM T52921 C8M4PI 70688696 Ki > 250 nM T52921 C3HAX5 70688697 Ki = 3.79 nM T52921 C7PNH3 70689062 Ki = 0.0373 nM T52921 CA3T1P 70689063 Ki = 0.127 nM T52921 CF7PZ4 70690755 Ki = 5.55 nM T52921 CMNL89 70690756 Ki = 128 nM T52921 CWB17N 70690757 Ki = 26.2 nM T52921 CX5VR6 70690758 Ki = 26.5 nM T52921 C8UYZ6 70690759 Ki > 250 nM T52921 CTB4I1 70690760 Ki = 0.96 nM T52921 CQJ6K3 70691171 Ki = 2.05 nM T52921 CEV6U7 70691173 Ki = 0.248 nM T52921 CY6E2Q 70691339 IC50 > 10000 nM T52921 C3E4FO 70692893 Ki = 101 nM T52921 CV61FR 70692894 Ki = 31.5 nM T52921 C05RKU 70692895 Ki = 286 nM T52921 CLM98A 70692896 Ki > 250 nM T52921 CU60IL 70694933 Ki > 250 nM T52921 CWO5F0 70695375 Ki = 0.169 nM T52921 CJ07AO 70696988 Ki > 250 nM T52921 C4Z0QA 70696990 Ki > 250 nM T52921 CV0P1X 70696991 Ki = 3.03 nM T52921 CFQ8Y9 70696992 Ki > 250 nM T52921 CTO0Y4 70697389 Ki = 0.458 nM T52921 CNE50L 70697390 Ki = 0.124 nM T52921 CG3U7F 70697391 Ki = 0.134 nM T52921 CEOQ43 71229805 Ki = 43.2 nM T52921 CJDR19 71230446 Ki = 44 nM T52921 CM0H5E 71454460 Ki = 22 nM T52921 CBEV63 71461579 Ki = 27.9 nM T52921 C0B7LC 71624265 Ki = 7.63 nM T52921 C7Q9VU 71624266 Ki = 15.26 nM T52921 CD9IO8 71624267 Ki = 212.8 nM T52921 CXZ6E1 71624268 Ki = 9.98 nM T52921 C0O6IR 71624269 Ki = 26.9 nM T52921 CW2G0T 71624270 Ki = 6.53 nM T52921 CBM1C8 71624387 Ki = 12.65 nM T52921 CML7K2 71624388 EC50 = 6.8 nM T52921 C1B9VM 71624389 Ki = 40.28 nM T52921 CWH6T3 72548703 IC50 = 0.98 nM T52921 CC6Q5R 72771081 Ki < 100 nM T52921 C7ZN1K 73345634 Ki = 0.05495 nM T52921 CN5S4A 73350483 Ki = 11.43 nM T52921 COS31U 73354624 Ki = 1700 nM T52921 CJQ25A 76309739 Ki = 4 nM T52921 CC01JG 76309740 Ki = 3 nM T52921 C69JCU 76313421 Ki = 31 nM T52921 CJR57Q 76313422 Ki = 401 nM T52921 CA4IN3 76313423 Ki = 16 nM T52921 CP3HV7 76313424 Ki = 10 nM T52921 CU56FN 76313425 Ki = 10 nM T52921 CPJ4N3 76313426 Ki = 36 nM T52921 C7LV2A 76313427 Ki = 13 nM T52921 CTN6G1 76316935 Ki = 15 nM T52921 C1AW8J 76316936 Ki = 22 nM T52921 CC2AG6 76316937 Ki = 17 nM T52921 CNAE72 76320663 Ki > 1000 nM T52921 CD0PC8 76320664 Ki > 1000 nM T52921 CF83DA 76320665 Ki = 6 nM T52921 C5W1XJ 76320666 Ki = 3 nM T52921 C0MI1G 76324308 Ki = 3 nM T52921 CI2A6W 76324309 Ki = 29 nM T52921 CT9XB8 76324310 Ki = 6 nM T52921 C4QM6R 76324311 Ki = 79 nM T52921 C6AY5S 76327872 Ki = 15 nM T52921 CCR5B1 76327873 Ki = 47 nM T52921 CL58DY 76327874 Ki = 9 nM T52921 CBVL29 76327875 Ki = 19 nM T52921 C64JDN 76327876 Ki = 7 nM T52921 C3G1LA 76327877 Ki = 42 nM T52921 CCN1M9 76331524 Ki = 75 nM T52921 CQ35XY 76331525 EC50 = 14 nM T52921 CDA37E 76335140 Ki = 72 nM T52921 CUZ30G 76335141 Ki = 122 nM T52921 CKZ7T2 76335142 Ki = 10 nM T52921 CQKT47 76335143 Ki = 10 nM T52921 C6K5RY 76335144 Ki = 10 nM T52921 CECO35 76335145 Ki = 12 nM T52921 CLH3X9 81689704 Ki = 80 nM T52921 CGH7J9 86279209 Ki = 3.16 nM T52921 C8HE3B 90306863 Ki = 4630 nM T52921 C1W9QL 90306885 Ki = 75 nM T52921 C1DOG7 90654745 Ki = 0.172 nM T52921 CX3WT1 90654746 Ki = 0.176 nM T52921 CC70MH 90654747 Ki = 0.145 nM T52921 C4ZQD5 90654748 Ki = 0.371 nM T52921 CBV23K 90654749 Ki = 0.114 nM T52921 C87NYV 90654750 Ki = 0.097 nM T52921 C20FOK 90654751 Ki = 0.105 nM T52921 CT91LC 90654752 Ki = 0.185 nM T52921 CT5U7G 90654753 Ki = 0.139 nM T52921 C42GMO 90654754 Ki = 0.0711 nM T52921 CBR5H7 90654755 Ki = 0.0954 nM T52921 C68VLU 90654756 Ki = 0.0648 nM T52921 C8GUX3 90654757 Ki = 0.122 nM T52921 C4Z6KQ 90654758 Ki = 0.0908 nM T52921 C13ACK 90654759 Ki = 0.0939 nM T52921 C7C5BM 90655970 Ki > 10000 nM T52921 CTV50C 90655971 Ki = 2.1 nM T52921 C1S5UB 90655972 Ki = 3.41 nM T52921 CV6A5T 90655973 Ki = 2.99 nM T52921 CL0D4Y 90655974 Ki = 8.63 nM T52921 C51CQN 90655975 Ki = 11.1 nM T52921 C2USA9 90655976 Ki = 76.6 nM T52921 CLKW80 90655977 Ki > 10000 nM T52921 C96DUE 90655978 EC50 = 72.2 nM T52921 C1N5QA 90655979 Ki > 10000 nM T52921 CK9FP8 90656664 Ki = 197 nM T52921 COGW86 90656666 Ki = 105 nM T52921 C9YKV8 90656667 Ki = 187 nM T52921 C3WLH8 90656668 Ki = 396 nM T52921 CP1ZW6 90663949 Ki > 5000 nM T52921 CZ9GL5 90663950 Ki = 45 nM T52921 CFK27M 90663951 Ki > 5000 nM T52921 CBT6F1 90663952 Ki > 5000 nM T52921 C1QAB3 90663953 Ki = 34 nM T52921 C07VRA 101341769 Ki = 39 nM T52921 C4VMI7 101354795 IC50 = 1.67 nM T52921 CBM3Q5 118662014 Ki = 68 nM T52921 CK8Y3E 118662042 Ki = 170 nM T52921 CS81PR 118662074 Ki = 0.8 nM T52921 C8AF6I 118662117 Ki = 29.5 nM T52921 CBJ16O 118662129 Ki = 1510 nM T52921 C4ZP0L 118662159 Ki = 1.6 nM T52921 CR6IU7 118662169 Ki = 2160 nM T52921 C7VE1O 118662183 Ki = 600 nM T52921 C1VR3B 118662189 Ki = 0.7 nM T52921 CG0R6H 118662291 Ki = 2.9 nM T52921 CI17PS 118662309 Ki = 5.8 nM T52921 CCIP14 118662342 Ki = 1.1 nM T52921 CB79UC 118662456 Ki = 2.3 nM T52921 C5LZ8I 118662460 Ki = 0.4 nM T52921 CM8TB4 118705898 Ki = 1300 nM T52921 C80UNO 118705899 Ki = 1500 nM T52921 C6RW0E 118705901 Ki = 880 nM T52921 C20RQZ 118711156 Ki = 1600 nM T52921 CV85YO 118711243 Ki = 5.4 nM T52921 CKUT03 118711485 Ki = 0.5 nM T52921 CI6BM7 118711486 Ki = 2 nM T52921 CMY0F1 118711490 Ki = 0.55 nM T52921 CMRV59 118711491 Ki = 1.1 nM T52921 CTVK82 118717442 IC50 = 1.39 nM T52921 CSIW96 118718262 Ki = 39 nM T52921 C4LM3W 118718263 Ki = 55 nM T52921 C2Q8YU 118718264 Ki = 116 nM T52921 C9BFP5 118718265 Ki = 5 nM T52921 CS14YZ 118718266 Ki = 7 nM T52921 CRBA23 118718267 Ki = 82 nM T52921 C4AS8L 118718268 Ki = 35 nM T52921 CP8I2K 118718269 Ki = 17 nM T52921 C6TGR8 118718270 Ki = 336 nM T52921 C3W1BL 118718271 Ki = 29 nM T52921 CPC23W 118718272 Ki = 24 nM T52921 C2Y4PK 118718273 Ki = 104 nM T52921 C8FC1Q 118718274 Ki = 4 nM T52921 C2BGR0 118718275 Ki = 27 nM T52921 CJZ1F7 118718276 Ki = 34 nM T52921 CCFR52 118718277 Ki = 15 nM T52921 C5O2VC 118718278 Ki = 58 nM T52921 CC0KE5 118718279 Ki = 7 nM T52921 CK1Q9B 118718280 Ki = 20 nM T52921 CB92OV 118718281 Ki = 50 nM T52921 CSK4N3 118718282 Ki = 173 nM T52921 CDBP05 118718283 Ki = 245 nM T52921 CDH69C 118718284 Ki = 670 nM T52921 CLRD02 118718285 Ki = 62 nM T52921 CYI4T2 118718286 Ki = 27 nM T52921 C2F8ZN 118718287 Ki = 99 nM T52921 CA9N0S 118718288 Ki = 11 nM T52921 CVT94Z 118718289 Ki = 6 nM T52921 C1RAX5 118718290 Ki = 10 nM T52921 CKNL94 118718291 Ki = 17 nM T52921 CKN54J 118718292 Ki = 20 nM T52921 CC6U5D 118718293 Ki = 210 nM T52921 C64JUV 118718294 Ki = 70 nM T52921 CICJ78 118718295 Ki = 68 nM T52921 CZMR06 118718296 Ki = 31 nM T52921 C92CER 118718297 Ki = 118 nM T52921 CP23YE 118718298 Ki = 50 nM T52921 COA69M 118718299 Ki = 39 nM T52921 CSW82H 118718300 Ki = 74 nM T52921 C2EGJ8 118718301 Ki = 11 nM T52921 CO5BV4 118718302 Ki = 12 nM T52921 CTF9L6 118722880 Ki = 7.4 nM T52921 CDI8J1 118722882 Ki = 0.5 nM T52921 C3T8YZ 118726261 IC50 = 61 nM T52921 C6I5HS 118726262 IC50 = 4.2 nM T52921 C10BIV 118726263 IC50 = 99.7 nM T52921 CA43CF 118726264 IC50 = 166 nM T52921 CLSG96 118726265 IC50 = 160 nM T52921 CYL40S 118726266 IC50 = 8 nM T52921 CPR0K2 118726267 IC50 = 14 nM T52921 CH9A3M 118726268 IC50 = 26 nM T52921 CEH89Y 118726269 IC50 = 3.9 nM T52921 CT7H2M 118726270 IC50 = 40.9 nM T52921 C1UD6R 118726271 IC50 = 8.8 nM T52921 CRK62Y 118726272 IC50 = 37 nM T52921 CF25IA 118726273 IC50 = 18 nM T52921 CQH1G3 118731120 Ki > 10000 nM T52921 CK0LH7 122179050 Ki = 97 nM T52921 CEY90C 122179051 Ki = 1270 nM T52921 CBP42W 122179052 EC50 = 14 nM T52921 CNCJ68 122179053 EC50 = 7.3 nM T52921 CY96XI 122179055 Ki = 820 nM T52921 C6LDU5 122179056 Ki = 240 nM T52921 C57GMN 122179057 Ki = 56 nM T52921 C0X6AF 122179058 Ki = 56 nM T52921 CS0B3O 122179059 Ki = 26 nM T52921 C09BYL 122179060 Ki = 47.8 nM T52921 CF83LN 122179061 Ki = 62.2 nM T52921 CC73XP 122179063 Ki = 571 nM T52921 C6YQM4 122179064 EC50 = 230 nM T52921 C9WF5T 122179567 EC50 = 323.59 nM T52921 CTA9E8 122179568 EC50 = 158.49 nM T52921 C35HVO 122179584 EC50 = 426.58 nM T52921 CF2W0K 122179586 EC50 = 208.93 nM T52921 CE3LH1 122179587 EC50 = 45.71 nM T52921 CAQ5B0 122409965 Ki = 0.53 nM T52921 C51MTO 124565311 Ki = 0.21 nM T52921 C1YEA7 127030671 Ki > 250 nM T52921 C1HO7F 127033703 Ki = 3.13 nM T52921 CB12AP 127033704 Ki > 250 nM T52921 C4NIU0 127034022 Ki = 5.65 nM T52921 C7ORD8 127034023 Ki = 5.55 nM T52921 CEWM81 127034292 Ki = 3.56 nM T52921 CBOC84 127034554 Ki = 18.1 nM T52921 CXMJ48 127043001 Ki = 27 nM T52921 CFU4H9 127043364 Ki = 47 nM T52921 C30BNK 127043559 Ki = 38 nM T52921 CCSZ68 127044528 Ki = 42 nM T52921 C1EHU5 129188443 Ki = 9.8 nM T52921 CD8FT9 129188454 Ki = 2.17 nM T52921 CC9Z0J 129188459 Ki = 10.3 nM T52921 CG57MT 134563466 Ki = 10.5 nM T52921 CE5RS7 134563496 Ki = 23.6 nM T52921 CAEY19 134563500 Ki = 216 nM T52921 C82SEF 134563650 Ki = 44.7 nM T52921 CC3HK6 134563655 Ki = 0.3 nM T52921 C4U9EM 134563691 Ki = 43.8 nM T52921 CFX37T 134563695 Ki = 129 nM T52921 CPEH72 134563698 Ki = 24.4 nM T52921 CR74XA 134563699 Ki = 31.8 nM T52921 C9PN6I 134578342 Ki = 15.9 nM T52921 CK62WY 134578456 Ki = 9.46 nM T52921 CN0C9Z 134578457 Ki = 1.47 nM T52921 C0HNI9 134578506 Ki = 64 nM T52921 C0JCQ2 134578518 Ki = 136 nM T52921 C1CH3X 135458466 IC50 = 199 nM T52921 CN14XB 136036819 Ki = 5.888 nM T52921 CL14DP 136043756 IC50 = 440 nM T52921 CC1N8P 136043758 IC50 > 1000 nM T52921 CUXY20 136043759 IC50 = 294 nM T52921 C7US0J 136043761 IC50 > 1000 nM T52921 CFLE34 136043762 IC50 > 1000 nM T52921 C0HPR7 136043764 IC50 > 1000 nM T52921 C9WN3S 136043765 IC50 = 580 nM T52921 CB5O8L 136043767 IC50 = 440 nM T52921 CW9HY3 136043768 IC50 > 1000 nM T52921 C8CTV4 136043771 IC50 = 140 nM T52921 CB36GF 136043772 IC50 > 1000 nM T52921 CIZ41F 136043774 IC50 > 1000 nM T52921 CKW90B 136043777 IC50 > 1000 nM T52921 CJL1Y8 136043778 IC50 > 1000 nM T52921 C5KZF8 136043779 IC50 = 58 nM T52921 C2LC8O 136043780 IC50 = 450 nM T52921 C9B0WD 136043781 IC50 = 568 nM T52921 CJM57B 136043782 IC50 = 233 nM T52921 C0A6NT 136043783 IC50 > 1000 nM T52921 C0QTA5 136043784 IC50 > 1000 nM T52921 CRGU10 136043785 IC50 > 1000 nM T52921 COL64J 136043786 IC50 = 120 nM T52921 CV5AJ0 136043787 IC50 > 1000 nM T52921 CH0VN9 136043788 IC50 = 62 nM T52921 C1GJE7 136043789 IC50 > 1000 nM T52921 CC8ZK4 136043790 IC50 = 210 nM T52921 C0QDL8 136043791 IC50 > 1000 nM T52921 CM2I3S 136043792 IC50 = 600 nM T52921 CZ6A5D 136043795 IC50 = 450 nM T52921 C24BXO 136043796 IC50 = 230 nM T52921 CQLF58 136043797 IC50 = 560 nM T52921 C9EF5P 136043798 IC50 > 1000 nM T52921 CEZ83O 136043799 IC50 > 1000 nM T52921 CFZX29 136043800 IC50 = 49 nM T52921 CVFX50 136043807 IC50 > 1000 nM T52921 C5TIE8 136043816 IC50 > 1000 nM T52921 C68CEZ 136043817 IC50 = 450 nM T52921 CCJ02K 136043818 IC50 > 1000 nM T52921 C06YGH 136043819 IC50 = 632 nM T52921 C1XV2U 136043820 IC50 > 1000 nM T52921 C53OLF 136043821 IC50 > 1000 nM T52921 C4NXF8 136043824 IC50 = 410 nM T52921 CX3H8P 146034954 EC50 = 72.44 nM T52921 C85LIH 146034955 EC50 = 7.244 nM T52921 CY5CL2 155521553 Ki = 20.9 nM T52921 CZ1V3B 155523994 IC50 = 0.63 nM T52921 CXH95L 155531153 Ki = 2.27 nM T52921 CTWG84 155533462 Ki = 2 nM T52921 C4RWI6 155536757 Ki = 27 nM T52921 CHJ59D 155537352 Ki = 15.5 nM T52921 C67WLH 155542684 Ki = 23.1 nM T52921 CU83VX 155544763 Ki = 11 nM T52921 CQ0GL3 155569552 Ki = 11 nM T52921 D00BIE 25084507 Ki = 0.34 nM T52921 D00HAJ 73347136 IC50 > 50000 nM T52921 D00LVW 44456141 IC50 = 3.42 nM T52921 D00XZH 44430025 Ki = 433 nM T52921 D00YCW 44426807 Ki = 19 nM T52921 D01CFO 44456028 IC50 = 7.42 nM T52921 D01MUV 10314141 Ki = 62 nM T52921 D01WMU 9820782 Ki = 4 nM T52921 D02NSY 10296561 Ki = 0.2399 nM T52921 D02TPK 44416445 IC50 = 0.0803 nM T52921 D02WBU 44456216 EC50 = 17.7 nM T52921 D03BVN 44456298 EC50 = 23.8 nM T52921 D03PTV 10022129 Ki = 59 nM T52921 D03UJW 22970051 Ki = 23 nM T52921 D04PUK 44426803 Ki = 613 nM T52921 D04WRO 44456337 IC50 = 218 nM T52921 D04ZQX 44426812 Ki = 18 nM T52921 D05NIE 44430036 Ki = 455 nM T52921 D05RII 44413409 Ki = 1140 nM T52921 D05YMD 44455999 IC50 = 21.3 nM T52921 D06MQG 44430018 Ki = 180 nM T52921 D06PHT 10269001 Ki = 13 nM T52921 D06PVO 44426806 Ki = 135 nM T52921 D06RSR 44456187 IC50 = 14.7 nM T52921 D07CIU 9924923 Ki = 55 nM T52921 D07FCB 9925737 Ki = 323 nM T52921 D07NMH 10093682 Ki = 51 nM T52921 D08BAW 44456185 IC50 = 1.86 nM T52921 D08DVV 44430026 Ki = 1147 nM T52921 D08IXN 5497186 Ki = 0.03 nM T52921 D08NDP 25080768 Ki = 0.1 nM T52921 D08QBS 44178080 IC50 = 4.6 nM T52921 D08QBU 44430029 Ki = 1667 nM T52921 D08TFY 10043439 Ki = 17 nM T52921 D08ZDP 44430014 Ki = 9155 nM T52921 D09BYD 20481138 Ki = 11 nM T52921 D09CTG 44416444 IC50 = 0.789 nM T52921 D09FJY 9863568 Ki = 2 nM T52921 D09KBQ 131534 Ki = 2151 nM T52921 D09LRO 44430008 Ki = 23 nM T52921 D09VRT 44426814 Ki = 16 nM T52921 D09XZM 10986104 IC50 = 3.03 nM T52921 D0A1XG 44416268 IC50 > 10000 nM T52921 D0A8NZ 44578000 Ki = 0.27 nM T52921 D0A8ZS 44456217 IC50 = 92.6 nM T52921 D0AC0A 10047612 Ki = 0.253 nM T52921 D0D0UP 10315818 Ki = 48 nM T52921 D0D9BB 10427620 Ki = 313 nM T52921 D0E3RQ 44416159 IC50 = 0.0464 nM T52921 D0F8AX 44430024 Ki = 376 nM T52921 D0F8CV 5462471 Ki > 10000 nM T52921 D0FF6S 16038374 IC50 > 10000 nM T52921 D0G4FA 10384734 Ki = 588 nM T52921 D0G7DF 44426827 Ki = 3 nM T52921 D0HN2M 44430609 Ki = 0.02818 nM T52921 D0IL9H 44430013 Ki = 1745 nM T52921 D0J5JO 44430009 Ki = 27 nM T52921 D0JH5D 44430007 Ki = 34 nM T52921 D0K2NY 44456101 IC50 = 5.67 nM T52921 D0L6QN 10070040 Ki = 24 nM T52921 D0L8YY 10066285 Ki = 5.7 nM T52921 D0M7TP 44456412 IC50 = 14.9 nM T52921 D0NE3U 5485199 IC50 > 10000 nM T52921 D0O7JV 44426810 Ki = 14 nM T52921 D0P3FP 44426808 Ki = 5 nM T52921 D0PN2C 44456140 IC50 = 2.81 nM T52921 D0PR2Q 44456220 EC50 = 27.6 nM T52921 D0Q2PO 25084509 Ki = 0.54 nM T52921 D0Q9TQ 10043898 Ki = 54 nM T52921 D0QH4A 10089987 Ki = 14 nM T52921 D0S2OA 10388166 Ki = 162 nM T52921 D0SE9S 9887077 Ki = 0.3 nM T52921 D0SN6V 44456299 EC50 = 46.5 nM T52921 D0T0GL 44456296 IC50 = 0.66 nM T52921 D0T4ZY 44426817 Ki = 134 nM T52921 D0T9KE 44430016 Ki = 85 nM T52921 D0TJ7R 97333 Ki = 1983 nM T52921 D0U6FM 44456339 IC50 = 21.7 nM T52921 D0V3OY 105104 Ki > 10000 nM T52921 D0VH3M 25088989 Ki = 0.83 nM T52921 D0W3VT 10091033 Ki = 24 nM T52921 D0W7CF 9963005 IC50 = 1.04 nM T52921 D0X4SX 10317947 Ki = 72 nM T52921 D0XX1Y 44426828 Ki = 53 nM T52921 D0Y0IE 44352919 EC50 = 1.97 nM T52921 D0Y2MT 44416158 IC50 = 11.6 nM T52921 D0Y4EW 6324645 EC50 = 0.3236 nM T52921 D0Y5LJ 10336926 Ki = 136 nM T52921 D0Y7KE 44430012 Ki = 1281 nM T52921 D0YM8F 25084510 Ki = 1.79 nM T52921 D0ZE2W 44430028 Ki = 2176 nM T98092 D02EEJ 6479267 Ki = 1.84 nM T98092 D0CE0O 11513676 Ki = 0.34 nM T98092 D0G7UX 5284373 Ki = 2.64 nM T98092 D0M2OY 53259809 Ki = 16800 nM T98092 D08MYL 6473876 Ki = 2.11 nM T98092 CY0Q4V 444384 IC50 = 2000000 nM T98092 CLYE08 497073 IC50 = 6000 nM T98092 C8SG7U 497075 IC50 > 10000000 nM T98092 CAWY91 497076 IC50 = 90000 nM T98092 CC9D3J 497077 IC50 > 10000000 nM T98092 CBMF04 497078 IC50 = 500000 nM T98092 C6KF5Y 1367020 IC50 = 580 nM T98092 CP61UY 2823177 IC50 = 920 nM T98092 CM6OW0 3190778 IC50 = 5.5 nM T98092 CDPT84 4128827 IC50 = 316 nM T98092 C7T6VH 4401642 IC50 = 14 nM T98092 CSQP36 5020377 IC50 = 303 nM T98092 CZ34OX 5116189 IC50 = 5500 nM T98092 C7DIT9 5493631 IC50 = 680000 nM T98092 C35VSF 5493632 IC50 = 1000000 nM T98092 CGN50H 5493634 IC50 = 260000 nM T98092 C8U3AT 5493635 IC50 = 115000 nM T98092 C5I2UC 5493638 IC50 = 280000 nM T98092 CNIC61 6475296 IC50 = 310 nM T98092 C8RA6C 6476061 IC50 = 11.1 nM T98092 CTXB32 6479257 IC50 = 3 nM T98092 CMH26D 6479258 IC50 = 47 nM T98092 C45EVU 6479259 IC50 = 15 nM T98092 CQ1X3C 6479260 IC50 = 61 nM T98092 C1YMW4 6479261 IC50 = 277 nM T98092 CAYZ53 6479262 IC50 = 97 nM T98092 CPCG74 6479263 IC50 = 128 nM T98092 C16CZK 6479264 IC50 = 19 nM T98092 CN1BF8 6479265 IC50 = 165 nM T98092 C8N4YK 6479266 IC50 = 110 nM T98092 CAGX82 6479268 IC50 = 6047 nM T98092 CM36KU 6479269 IC50 = 1572 nM T98092 CJWU53 6479270 IC50 = 882 nM T98092 CRV94O 6479271 IC50 = 959 nM T98092 C03LTJ 10034324 IC50 = 934 nM T98092 CODJ10 10626583 Ki = 795 nM T98092 CO9XA6 10819131 IC50 = 1500000 nM T98092 CF45ID 11516665 IC50 = 20 nM T98092 CGP87C 11531251 IC50 = 951 nM T98092 CSY31B 11559871 IC50 = 748 nM T98092 C6M1ZU 11567780 IC50 = 320 nM T98092 CJ27OG 11588606 IC50 = 140 nM T98092 CN8M2B 11617502 IC50 = 71 nM T98092 CS2Y6M 11631957 IC50 = 60 nM T98092 CX63ZC 11632684 IC50 = 60 nM T98092 CLP34W 11638938 IC50 = 592 nM T98092 CS3YJ8 11660364 IC50 = 640 nM T98092 C37WLM 11675245 IC50 = 528 nM T98092 C3SK8D 11703833 IC50 = 880 nM T98092 C2QN6F 11710570 IC50 = 1437 nM T98092 C73OMC 11717355 IC50 = 458 nM T98092 C89EKB 11718015 IC50 = 499 nM T98092 CUY92Q 13422114 IC50 = 130 nM T98092 CC6XY7 13578707 IC50 = 350 nM T98092 C8KA7W 20415061 IC50 = 460 nM T98092 C31GDL 24814873 IC50 = 14 nM T98092 C2ON4L 25044910 IC50 = 690 nM T98092 CY8HB6 25046022 IC50 = 330 nM T98092 CT2E3I 25098032 IC50 = 590 nM T98092 CK0P2Q 42630203 IC50 = 650 nM T98092 C69CNK 44248910 IC50 > 10000 nM T98092 C46XEC 44248911 IC50 = 103 nM T98092 CS6N9K 44248912 IC50 = 71.2 nM T98092 CHX9S4 44248913 IC50 = 159 nM T98092 CSDG42 44248914 IC50 > 10000 nM T98092 CJT1A8 44249039 IC50 = 364 nM T98092 CVW1T9 44249040 IC50 = 263 nM T98092 CNFI87 44249041 IC50 = 2.59 nM T98092 CW6LT7 44249042 IC50 = 1.52 nM T98092 C7U6PN 44249044 IC50 = 1910 nM T98092 C1HPV8 44249170 IC50 > 10000 nM T98092 CW4AU3 44249173 IC50 = 12.1 nM T98092 CKO3I0 44249174 IC50 > 10000 nM T98092 CL7M2J 44249303 IC50 = 620 nM T98092 C97JUQ 44249304 IC50 > 10000 nM T98092 C0SVJ1 44249305 IC50 = 31.6 nM T98092 CA3K2N 44249306 IC50 > 10000 nM T98092 CBEL85 44249307 IC50 = 370 nM T98092 C5M4VW 44249309 IC50 = 136 nM T98092 CR2K7N 44249310 IC50 > 10000 nM T98092 C57MCG 44249414 IC50 > 10000 nM T98092 CSJD94 44249415 IC50 > 10000 nM T98092 CER54N 44294512 IC50 = 2500000 nM T98092 CKYA61 44294584 IC50 = 850000 nM T98092 C4R1DL 44294708 IC50 > 10000000 nM T98092 CTE19D 44294709 IC50 > 10000000 nM T98092 CT5IJ4 44294814 IC50 = 2800000 nM T98092 C4GLS0 44294838 IC50 = 760000 nM T98092 C5EQ7U 44295020 IC50 = 1300000 nM T98092 CHI01J 44295050 IC50 = 1500000 nM T98092 CS5I9W 44295136 IC50 = 970000 nM T98092 COCG50 44295258 IC50 = 820000 nM T98092 CV7PD8 44341483 IC50 = 48 nM T98092 C5M1FB 44341507 IC50 = 256 nM T98092 CM9L8P 44365970 IC50 = 1500000 nM T98092 C50FPJ 44366040 IC50 = 2500000 nM T98092 C0JKL6 44366208 IC50 = 2600000 nM T98092 C98VGM 44366209 IC50 = 165000 nM T98092 C6PCZ9 44366232 IC50 = 850000 nM T98092 CRES48 44366233 IC50 = 325000 nM T98092 C7AQ3R 44366260 IC50 = 2100000 nM T98092 CS74HY 44366261 IC50 = 970000 nM T98092 CEH4W6 44366303 IC50 = 820000 nM T98092 CF3B2I 44366350 IC50 = 260000 nM T98092 C0I3BR 44366351 IC50 = 760000 nM T98092 C9HQ5S 44366390 IC50 = 2800000 nM T98092 CY89LF 44366391 IC50 = 1300000 nM T98092 CDJ21S 44366404 IC50 = 500000 nM T98092 CPW1A7 44366405 IC50 = 90000 nM T98092 C4SQ1N 44366450 IC50 = 280000 nM T98092 CUI2X6 44366451 IC50 = 6000 nM T98092 CMCP73 44366452 IC50 = 365000 nM T98092 C2LG1F 44366453 IC50 = 115000 nM T98092 C5Q4VN 44393426 Ki = 100 nM T98092 CP57YU 44393427 Ki = 75 nM T98092 CGX7M4 44393512 Ki = 10 nM T98092 CGP76Z 44393513 Ki = 24 nM T98092 CU0RC4 44393514 Ki = 18 nM T98092 CZAD42 44406917 IC50 = 4100 nM T98092 C0FLH5 44582698 IC50 = 740 nM T98092 C0ON5I 44582699 IC50 = 810 nM T98092 CW3R7N 44582757 IC50 = 740 nM T98092 CCV89D 44582780 IC50 = 880 nM T98092 CZM71K 44582804 IC50 = 600 nM T98092 CWF96D 44582805 IC50 = 450 nM T98092 CYN7C5 44582823 IC50 = 160 nM T98092 CW4P8K 44582824 IC50 = 450 nM T98092 CX94NI 45138814 IC50 = 2.4 nM T98092 CN72XD 45269870 IC50 > 10000 nM T98092 CS30FH 49863381 IC50 = 206 nM T98092 C3YI2V 49863382 IC50 = 950 nM T98092 CS48JU 49863383 IC50 = 4.75 nM T98092 CWI47U 50899161 IC50 = 26.6 nM T98092 CHN71J 52940634 IC50 = 31.2 nM T98092 CQ83LE 52940669 IC50 = 22.9 nM T98092 C2H0IK 52940670 IC50 = 46 nM T98092 CPKZ45 52940671 IC50 = 35.2 nM T98092 C7MA9P 52941831 IC50 = 9.12 nM T98092 CH9QA8 52941859 IC50 = 21.4 nM T98092 C97YWD 52945243 IC50 = 26.7 nM T98092 CE05IO 52945473 IC50 = 218 nM T98092 C43LWJ 52945496 IC50 = 140 nM T98092 C3BCG7 52946681 IC50 = 83.5 nM T98092 CR63JF 52946682 IC50 = 22.8 nM T98092 CH8TZ9 52946683 IC50 = 103 nM T98092 C7KW3U 52947912 IC50 = 23 nM T98092 C4KAU1 52947949 IC50 = 662 nM T98092 CGX04A 52947950 IC50 = 65.2 nM T98092 CS90AU 52952820 IC50 = 33.11 nM T98092 CBWK59 53321090 Ki = 106 nM T98092 CNS79R 53344622 IC50 = 2.7 nM T98092 CPD19A 53357115 IC50 = 350 nM T98092 CMYW90 53357116 IC50 = 630 nM T98092 C75LWY 53357117 IC50 = 500 nM T98092 C40GVQ 53357247 IC50 = 360 nM T98092 CC0Y1S 53357248 IC50 = 390 nM T98092 CPM2F7 53357386 IC50 = 330 nM T98092 COP18F 53357507 IC50 = 520 nM T98092 C4P3GC 53357508 IC50 = 420 nM T98092 C4O0YX 53357509 IC50 = 4.1 nM T98092 C96CAE 53357630 IC50 = 450 nM T98092 C8C9ZH 53358962 IC50 = 1.1 nM T98092 C3VJ0N 56668120 IC50 = 2000000 nM T98092 C30PVF 56675024 IC50 = 2600000 nM T98092 CFMP72 56678333 IC50 = 2100000 nM T98092 CFAY29 56678334 IC50 = 165000 nM T98092 CQB1I0 57384849 Ki = 14 nM T98092 CZK8P2 57384850 Ki = 65 nM T98092 CX67HU 57385085 Ki = 4 nM T98092 C6PXU0 57398046 IC50 = 4.9 nM T98092 C6ZK4A 67978739 Ki = 16 nM T98092 C6RT1L 71590783 IC50 = 740 nM T98092 CC0TY2 71590784 IC50 = 810 nM T98092 CH23LT 71596756 IC50 = 550 nM T98092 CZOT97 71596824 IC50 = 380 nM T98092 CC37ZO 71596825 IC50 = 330 nM T98092 C2IJ6X 71596826 IC50 = 460 nM T98092 CSE28O 73333514 Ki = 23 nM T98092 CDF54U 73333515 Ki = 10.7 nM T98092 CKS08Z 73333613 Ki = 12.4 nM T98092 C5FWY3 73333614 Ki = 43.9 nM T98092 C2LR7I 73333729 Ki = 11.8 nM T98092 CQH16I 73333730 Ki = 36.6 nM T98092 CRA39X 73333846 Ki = 57.7 nM T98092 C47PVY 73347049 IC50 = 680000 nM T98092 CKV1A9 73348786 IC50 = 2.3 nM T98092 CIXM26 73353051 IC50 = 16 nM T98092 C5J6GK 122437357 IC50 = 11.2 nM T98092 CUKL46 127038149 IC50 = 10000 nM T98092 CF7KS5 127038150 IC50 = 10000 nM T98092 C6HPE3 127038151 IC50 = 10000 nM T98092 CQC1L7 127038489 IC50 = 940 nM T98092 CI8EO6 127039060 IC50 = 10000 nM T98092 C7NW5Q 127039075 IC50 = 2760 nM T98092 CSU85H 127039831 IC50 = 10430 nM T98092 CA1P8V 127039832 IC50 = 10260 nM T98092 C2JQ4V 127039851 IC50 = 10000 nM T98092 C1DTR2 127039852 IC50 = 1220 nM T98092 CI03BD 127040172 IC50 = 10800 nM T98092 C0OTQ9 127040173 IC50 = 10000 nM T98092 CA75UB 127040174 IC50 = 10000 nM T98092 CC0GN1 127040175 IC50 = 10000 nM T98092 C8PI2G 127041686 IC50 = 10000 nM T98092 CS0EM4 127041788 IC50 = 10330 nM T98092 CE0KL8 127041789 IC50 = 10000 nM T98092 C35DGM 127042320 IC50 = 11620 nM T98092 C2VGI1 136220121 Ki = 64.7 nM T98092 C2ZA8L 137348679 Ki = 7 nM T98092 CY46VP 137637353 Ki = 4.3 nM T98092 D04PGW 6475368 IC50 = 166 nM T98092 D07ABJ 44358392 IC50 = 783 nM T98092 D07IQR 11639129 IC50 = 361 nM T98092 D0P6TX 3663276 IC50 = 754 nM T98092 D0X5JR 11574097 IC50 = 810 nM T52638 D03LWG 53235510 IC50 > 10000 nM T52638 D07EHV 44814409 IC50 > 10000 nM T52638 D0E3TC 44259 IC50 = 12100 nM T52638 C1ZPA9 1292979 IC50 = 623 nM T52638 C1XS2J 54760383 IC50 > 10000 nM T52638 CV63UL 67240318 IC50 > 10000 nM T52638 CM8LU3 122177129 IC50 = 420 nM T52638 CU5V7A 129318960 IC50 = 39 nM T52638 C38TVL 129318961 IC50 = 750 nM T52638 CX48MD 133080583 EC50 = 352 nM T52638 CTR4A0 135383414 IC50 = 95 nM T52638 C8MY4I 137632407 IC50 = 60 nM T52638 CTKX07 137635009 IC50 = 971 nM T52638 CLK3Y7 137635621 IC50 = 106 nM T52638 C0IMX2 137642056 Ki = 32.43 nM T52638 CVR5C8 137654407 IC50 = 2140 nM T52638 CLMT19 137660903 IC50 = 6 nM T52638 C2MD1Q 155513187 IC50 > 10000 nM T52638 D06HVH 54613583 IC50 > 10000 nM T56556 D00YZD 54726191 IC50 = 67000 nM T56556 D04AIT 5280445 IC50 = 8900 nM T56556 D07BSQ 5994 IC50 = 125892.54 nM T56556 D07POC 176870 IC50 = 50000 nM T56556 D09XZB 123631 IC50 = 1100 nM T56556 D0AZ3C 5291 IC50 = 4897.79 nM T56556 D0BP9C 193962 IC50 = 6000 nM T56556 D0J4JM 5770 IC50 = 12600 nM T56556 D0K8KX 5280343 EC50 = 30 nM T56556 D0OB1J 39186 IC50 = 851138.04 nM T56556 D0Q0PR 54675769 IC50 = 104000 nM T56556 D0R0FE 2520 EC50 = 900 nM T56556 D0R3JB 4212 IC50 = 903.8 nM T56556 D0T0KA 4474 IC50 = 16595.87 nM T56556 D01GFX 11640390 EC50 = 104 nM T56556 D02HTD 25167947 IC50 = 1400 nM T56556 D02QWY 24785538 IC50 = 10200 nM T56556 D0CE0O 11513676 IC50 = 2500 nM T56556 D0G7UX 5284373 EC50 = 1750 nM T56556 D0J1HB 23063810 IC50 = 65400 nM T56556 D0L4FS 5280961 IC50 = 6900 nM T56556 D00OWF 5280953 IC50 = 5080 nM T56556 D04RLX 148201 EC50 = 10 nM T56556 D09FGX 119373 IC50 = 400 nM T56556 D0Q7HO 4705 IC50 = 1730 nM T56556 C4DS3F 2361 IC50 = 6050 nM T56556 CQ9MW6 68077 IC50 = 17000 nM T56556 CJ65ZE 72344 IC50 = 4900 nM T56556 CSHM20 73201 IC50 = 8900 nM T56556 CI5UP7 88881 IC50 = 9200 nM T56556 C5ZCH7 97332 IC50 = 1880 nM T56556 CL97OF 97548 IC50 = 1280 nM T56556 CD8L6K 97696 IC50 = 7900 nM T56556 C6I9HU 97860 IC50 = 19000 nM T56556 C3NC7T 114429 IC50 = 11000 nM T56556 C8NLJ2 145659 IC50 = 8300 nM T56556 CNVB16 146013 IC50 = 1280 nM T56556 C4FEY6 147157 IC50 = 3400 nM T56556 C7E5NC 150893 IC50 = 1400 nM T56556 C4J5ZF 185617 IC50 = 10000 nM T56556 CRE67B 265724 IC50 = 1010 nM T56556 CABJ72 276138 IC50 = 1230 nM T56556 C1Q0WH 281852 IC50 = 1690 nM T56556 CPF26C 324081 IC50 = 10700 nM T56556 C4VJH5 324094 IC50 = 16600 nM T56556 CMC10D 324099 IC50 = 9000 nM T56556 CP5B4K 369597 IC50 = 4900 nM T56556 CKC6U2 369599 IC50 = 2800 nM T56556 CO6AM3 378567 IC50 = 17000 nM T56556 CA9IM5 396723 IC50 = 860 nM T56556 CVN3Z5 403923 IC50 = 451 nM T56556 C5YX1H 406017 IC50 = 30000 nM T56556 CHP8G0 406584 IC50 = 960 nM T56556 CWXZ47 406585 IC50 = 15000 nM T56556 CL6QB8 407032 IC50 = 4800 nM T56556 CC1Q8J 409920 IC50 = 6300 nM T56556 C3YG0Z 436659 IC50 > 20000 nM T56556 CWZ14N 468116 IC50 > 20000 nM T56556 CMT3P0 480764 IC50 = 3100 nM T56556 CL6E7C 609712 IC50 = 10000 nM T56556 C14NHZ 624831 IC50 = 12400 nM T56556 C34KNT 631171 IC50 = 2140 nM T56556 CSA18D 651672 IC50 = 940 nM T56556 C90LPE 688666 IC50 = 6500 nM T56556 CMR6U0 693195 IC50 = 2630 nM T56556 CH0DT9 693197 IC50 = 150 nM T56556 C1NZL9 693198 EC50 = 72 nM T56556 CW2U6N 698956 IC50 = 130 nM T56556 C19VMW 698960 EC50 = 72 nM T56556 C65SGT 712193 IC50 = 645 nM T56556 CH6MV7 715632 IC50 = 6380 nM T56556 C2NI7K 718862 IC50 = 890 nM T56556 CNS78D 719277 IC50 = 1150 nM T56556 CST9W8 719279 IC50 = 1480 nM T56556 CEC0X3 719282 IC50 = 2250 nM T56556 CRX4Q5 719284 IC50 = 1930 nM T56556 C6AKG9 735124 IC50 = 8120 nM T56556 C8OB6U 787509 EC50 = 50 nM T56556 C64RUF 877998 EC50 = 70 nM T56556 CXR0P5 917533 IC50 = 15800 nM T56556 C2X8PT 930478 IC50 = 108 nM T56556 CXQ4P8 1183964 IC50 = 944 nM T56556 CB31HC 1186125 IC50 = 362 nM T56556 CM42KO 1187243 IC50 = 107.15 nM T56556 CYT7E4 1214451 EC50 = 13 nM T56556 CCNX23 1361994 IC50 = 216 nM T56556 C35OEM 1413870 IC50 = 28900 nM T56556 CV7F8O 1418188 IC50 = 405 nM T56556 CAXQ59 1424290 IC50 = 2780 nM T56556 C2FL5J 1553837 IC50 = 250 nM T56556 C5RA6J 1566118 IC50 = 166 nM T56556 CQYO27 1597005 IC50 = 10700 nM T56556 C0M7DO 1696333 IC50 = 1340 nM T56556 COAE97 2176800 IC50 = 1060 nM T56556 C6ZFC1 2463411 IC50 = 791 nM T56556 CG3V9C 2549745 IC50 = 224 nM T56556 C2ZDU4 2562583 IC50 = 570 nM T56556 CFC30O 2789499 EC50 = 11 nM T56556 C01JRM 3034694 IC50 = 9300 nM T56556 C69NQO 3627000 EC50 = 58 nM T56556 C72VLI 4022553 IC50 = 196 nM T56556 C43JKM 4271896 IC50 = 3860 nM T56556 CHV3N6 4786429 IC50 = 360 nM T56556 CKG0Q7 4839583 IC50 = 724 nM T56556 CGKX02 4841865 IC50 = 1320 nM T56556 CN35MZ 4970131 IC50 = 11800 nM T56556 C8PN0C 5280682 IC50 = 680 nM T56556 CF6KZ2 5281677 IC50 = 17200 nM T56556 CQ9GX3 5320462 IC50 = 2000 nM T56556 C2TVO1 5328202 IC50 = 1980 nM T56556 C0O4SM 5332516 IC50 = 2630 nM T56556 CI6TE3 5348770 IC50 = 9230 nM T56556 CTO51S 5352005 IC50 = 540 nM T56556 CQL05G 5355469 IC50 = 3000 nM T56556 CTPE71 5355684 IC50 = 3280 nM T56556 CN8GP9 5355845 IC50 = 16200 nM T56556 C9T0DZ 5355846 IC50 = 10500 nM T56556 CW1UM5 5357488 IC50 = 2200 nM T56556 CU29TR 5373259 IC50 = 530 nM T56556 CV7Z2A 5373273 IC50 = 1060 nM T56556 CRW09S 5373997 IC50 = 3090 nM T56556 C09NZD 5380645 IC50 = 31020 nM T56556 C2KZF0 5476176 IC50 = 2400 nM T56556 CO17YB 5702790 IC50 = 1730 nM T56556 CI4U9Z 5711223 IC50 = 12050 nM T56556 CVF14X 5712116 IC50 = 4970 nM T56556 CCAT78 5723044 IC50 = 2190 nM T56556 CR51QS 5729243 IC50 = 22390 nM T56556 CG25KB 5729341 IC50 = 1950 nM T56556 CE0W8M 5730384 IC50 = 7800 nM T56556 CD18KY 5730712 EC50 = 2100 nM T56556 CA9WL4 5797184 IC50 = 18200 nM T56556 C7LKC3 5822497 IC50 = 10720 nM T56556 C29JCA 5909266 IC50 = 3320 nM T56556 CDLV62 5936200 IC50 = 2200 nM T56556 C9DB2C 5953849 IC50 = 850 nM T56556 CG82WY 5978982 IC50 = 2820 nM T56556 CFO1R0 6063342 IC50 = 1910 nM T56556 CP8O7I 6070899 IC50 = 1470 nM T56556 CMC06O 6123891 IC50 = 6440 nM T56556 C90ACD 6199559 IC50 = 9830 nM T56556 CYX45A 6213016 IC50 = 4910 nM T56556 CV91FR 6213967 EC50 = 1250 nM T56556 C6SZW5 6229071 IC50 = 7290 nM T56556 CU3X5P 6229072 IC50 = 9210 nM T56556 CFO9D1 6256073 IC50 = 8700 nM T56556 CX87NG 6475921 IC50 = 12300 nM T56556 COF72V 6919145 IC50 = 910 nM T56556 C0MGV7 7048595 IC50 = 3790 nM T56556 CNH60W 7946188 IC50 = 7220 nM T56556 C0O7PG 9109771 IC50 = 810 nM T56556 CLIG51 9281828 IC50 = 753 nM T56556 C1IPS5 9283400 EC50 = 85 nM T56556 C0D2SZ 9448204 IC50 = 4280 nM T56556 C4CF5U 9448550 EC50 = 512 nM T56556 C40XDF 9880195 EC50 = 14 nM T56556 CHI5S9 9975676 IC50 = 5910 nM T56556 C26IPN 10047854 IC50 = 5700 nM T56556 CY73KI 10322450 IC50 = 4 nM T56556 C7QYK3 10359377 IC50 = 830 nM T56556 C7Z8IW 10379829 IC50 = 4250 nM T56556 C0V5QI 10394010 IC50 = 11000 nM T56556 CT9MP2 10404096 IC50 = 3800 nM T56556 C36PIN 10407830 IC50 = 8190 nM T56556 C78HZG 10495050 IC50 = 6160 nM T56556 CR9SE7 10540319 IC50 = 6370 nM T56556 CEZ2B4 10612087 IC50 = 1940 nM T56556 CIOL78 10699195 IC50 = 16000 nM T56556 CF1UM5 10746774 IC50 = 29000 nM T56556 CI1RC8 10830017 IC50 = 9100 nM T56556 CT8PY0 10899903 IC50 > 20000 nM T56556 CDX92T 11210677 IC50 = 2460 nM T56556 CL1YX5 11246927 IC50 = 3620 nM T56556 C0SO6D 11312797 IC50 = 930 nM T56556 CL3YO1 11537442 IC50 = 700 nM T56556 C2C3WI 11957988 IC50 = 2089.3 nM T56556 C47ZJY 11996857 IC50 = 20000 nM T56556 CR3X7L 12388142 IC50 = 2890 nM T56556 C0KZQ2 12388145 IC50 = 5210 nM T56556 CS4YL1 12511782 IC50 = 2140 nM T56556 CRE67S 12753643 IC50 = 2580 nM T56556 CT24DO 13147509 IC50 = 920 nM T56556 C5VXB4 13147512 IC50 = 3550 nM T56556 C4GZ8Y 13168110 EC50 = 41 nM T56556 C5X4VH 13250463 IC50 > 20000 nM T56556 CM28RZ 13329020 IC50 = 424 nM T56556 C1U9IN 13707046 IC50 = 2890 nM T56556 C5DMA3 14034811 IC50 = 260 nM T56556 CRIH25 14259001 IC50 = 6600 nM T56556 CG0ZK1 14531326 EC50 = 900 nM T56556 C2LA5S 15556477 IC50 = 5680 nM T56556 CJ78CV 15648569 IC50 = 720 nM T56556 CJ5XV3 15965811 IC50 > 100000 nM T56556 C19FNV 15993184 EC50 = 12 nM T56556 CLD92G 15999199 EC50 = 4.7 nM T56556 C0A3IV 16092354 IC50 = 1190 nM T56556 C3TH4N 16092356 IC50 = 689 nM T56556 C7DW6Y 16092357 EC50 = 131 nM T56556 C7TBI5 16339054 IC50 = 15400 nM T56556 CMVW98 16618023 EC50 = 1310 nM T56556 CD04RW 16745324 IC50 = 2500 nM T56556 CN73EP 16805556 IC50 = 4790 nM T56556 CPOZ18 17375361 IC50 = 11200 nM T56556 CX06NR 17412108 IC50 = 16000 nM T56556 C5MOF7 17497142 IC50 = 10400 nM T56556 COG12F 17585222 IC50 = 8680 nM T56556 CPE15U 18004103 IC50 = 14500 nM T56556 CYSV63 19392346 IC50 = 60000 nM T56556 C3UT8G 20239593 IC50 = 170 nM T56556 CJ4Z1L 20646908 IC50 = 20900 nM T56556 C59FWO 20646970 IC50 = 51300 nM T56556 CIZV45 20646979 IC50 = 40000 nM T56556 CB7T2K 20963109 EC50 = 1.2 nM T56556 C2RQF6 21002393 IC50 = 1180 nM T56556 CB50QE 21418982 IC50 = 648 nM T56556 CCJ3M5 22004538 IC50 = 32400 nM T56556 CFI13S 22310708 IC50 = 420 nM T56556 CDQX04 22330280 IC50 = 462 nM T56556 C9IHU3 22330507 IC50 = 1990 nM T56556 C85SLA 23792651 IC50 = 8900 nM T56556 C7TOB4 23906108 IC50 = 1660 nM T56556 CU1G8A 23940255 IC50 = 87.1 nM T56556 CRCA82 23965087 EC50 = 21 nM T56556 CX2UF8 24016488 IC50 = 612 nM T56556 C2XB8M 24017959 IC50 = 183 nM T56556 C3ESV6 24178402 EC50 = 90000 nM T56556 C6AU1C 24204512 IC50 = 790 nM T56556 CU7LR8 24208774 IC50 = 458 nM T56556 CLY6U7 24626581 IC50 = 921 nM T56556 CCPS81 24764502 IC50 = 35000 nM T56556 CKW04J 24807980 EC50 = 7000 nM T56556 CJUW92 24807981 EC50 = 1500 nM T56556 CP8H2D 24807987 EC50 = 58000 nM T56556 C9T7BZ 24808155 EC50 = 75000 nM T56556 C9SMO0 24808156 EC50 = 120000 nM T56556 CW4EM8 24808157 EC50 = 150000 nM T56556 C7UV4H 24808344 EC50 = 500 nM T56556 C9F8CE 24826109 IC50 = 430 nM T56556 C9LXA0 24827935 IC50 = 350 nM T56556 C39SHG 24882446 IC50 = 23988.33 nM T56556 CF1JU8 24978503 IC50 = 230 nM T56556 C60EJI 25113688 EC50 = 73000 nM T56556 CS3ZN9 25195356 IC50 = 350 nM T56556 C2YA4G 25217469 IC50 = 1750 nM T56556 CM80XH 25222999 IC50 = 60 nM T56556 CSRV83 25223000 IC50 = 172 nM T56556 C26ZQR 25223001 IC50 = 632 nM T56556 C0S7AF 25223002 IC50 = 317 nM T56556 CZ4A5K 25223105 IC50 = 858 nM T56556 CKY89F 25223106 IC50 = 1990 nM T56556 CIJU21 25223199 IC50 = 119 nM T56556 CUZ5S9 25223200 IC50 = 183 nM T56556 C03FQV 25223201 IC50 = 552 nM T56556 C8S6UH 25223298 IC50 = 1015 nM T56556 CZQE36 25223299 IC50 = 977 nM T56556 C6O2ZR 25225119 EC50 = 30000 nM T56556 C8W9VD 25249649 IC50 > 10000 nM T56556 C78LKG 26213315 IC50 = 4100 nM T56556 CJPM47 31538107 IC50 = 1350 nM T56556 CI4AK1 39969954 IC50 = 14400 nM T56556 C0X8OT 44221093 IC50 = 10200 nM T56556 C9BNA1 44248179 EC50 = 63.2 nM T56556 C4DBF9 44257640 IC50 = 5900 nM T56556 C2NK1G 44428701 IC50 = 770 nM T56556 C4NCQ7 44428711 IC50 > 20000 nM T56556 CUIG60 44428712 IC50 = 450 nM T56556 CQ6A3K 44428713 IC50 = 560 nM T56556 CNBA28 44428714 IC50 = 1380 nM T56556 C43CIH 44451513 IC50 = 77624.71 nM T56556 CMHP85 44451563 IC50 = 263026.8 nM T56556 C29SBO 44451564 IC50 = 6606.93 nM T56556 C1G2CB 44451590 IC50 = 7585.78 nM T56556 C6NW0Q 44451617 IC50 = 14454.4 nM T56556 C1ENZ0 44451645 IC50 = 44668.36 nM T56556 CB0OL9 44451671 IC50 = 6025.6 nM T56556 CC9LK5 44451719 IC50 = 6025.6 nM T56556 CS4RX9 44451745 IC50 = 7244.36 nM T56556 C9Z4VY 44451773 IC50 = 12882.5 nM T56556 CTP09O 44451801 IC50 = 11481.54 nM T56556 CP69AF 44451832 IC50 = 22908.68 nM T56556 C45VCM 44451857 EC50 = 15000 nM T56556 C4T5UP 44451866 IC50 = 21877.62 nM T56556 CI1Y5L 44451888 IC50 = 64565.42 nM T56556 CP3B8R 44451889 IC50 = 36307.81 nM T56556 C3S5OK 44451912 IC50 = 5011.87 nM T56556 C6M3ZN 44451913 IC50 = 47863.01 nM T56556 C9AOQ4 44562411 IC50 = 15135.61 nM T56556 CLBO81 44565459 IC50 = 9080 nM T56556 C7NRZ8 44565460 IC50 = 6760 nM T56556 CN03BJ 44565480 IC50 = 2610 nM T56556 C38FXL 44565481 IC50 = 58400 nM T56556 CZUI80 44565482 IC50 = 74100 nM T56556 CZT54M 44565509 IC50 = 74100 nM T56556 C4Q2ER 44593438 IC50 = 24547.09 nM T56556 CE6F2U 45272659 IC50 = 22600 nM T56556 COPA25 46227750 IC50 = 10200 nM T56556 COA30H 46227751 IC50 = 630 nM T56556 CLWR13 46227752 IC50 = 500 nM T56556 C54HFY 46232422 IC50 > 100000 nM T56556 C5TJ4Y 46232423 IC50 = 25200 nM T56556 CY2RN7 46232494 IC50 > 100000 nM T56556 CW9J2R 46232495 IC50 > 100000 nM T56556 CO7V0S 46232496 IC50 > 100000 nM T56556 CZ89LA 46232497 IC50 = 15400 nM T56556 C4RUB7 46232498 IC50 = 6400 nM T56556 CR96LU 46232536 IC50 = 18800 nM T56556 C6UW4G 46232537 IC50 = 11100 nM T56556 C5ATF2 46232538 IC50 = 23200 nM T56556 CKXH76 46232539 IC50 > 100000 nM T56556 CXI72Q 46359934 IC50 = 1430 nM T56556 C0L6DC 46359963 IC50 = 60 nM T56556 CD64QE 49816175 IC50 = 1270 nM T56556 C72QDG 49844541 IC50 = 8920 nM T56556 CY4XL9 50806112 IC50 = 1890 nM T56556 C5PHF6 51041756 IC50 = 15500 nM T56556 C5M9DP 51041990 IC50 = 8400 nM T56556 CL29IG 53321447 IC50 = 6500 nM T56556 CPL41H 54341571 IC50 = 13600 nM T56556 C4Z7MF 54580539 IC50 > 100000 nM T56556 C96NWY 54580541 IC50 > 6200 nM T56556 CN30LW 54581539 IC50 > 5000 nM T56556 C6AIG3 54582535 IC50 = 183 nM T56556 CY24RJ 54582627 IC50 = 508 nM T56556 CN38OK 54583506 IC50 > 50000 nM T56556 CLTM38 54586400 IC50 > 50000 nM T56556 CK52PH 54586413 IC50 = 130 nM T56556 CIAU38 54587418 IC50 > 50000 nM T56556 CKZ01T 54587433 IC50 = 390 nM T56556 CB4DX1 54754510 IC50 = 450 nM T56556 CS7XP1 54754512 IC50 = 350 nM T56556 C4WO8B 56681840 IC50 = 270 nM T56556 C1H9ML 56764960 IC50 = 1390 nM T56556 C5EN2Q 56924700 IC50 = 170 nM T56556 CTX1N3 56924701 EC50 = 31 nM T56556 CP1VK5 56951135 IC50 = 16300 nM T56556 C2SF8B 56951136 IC50 = 470 nM T56556 C2KMN3 56951137 IC50 = 180 nM T56556 CAT80Q 56951138 IC50 = 200 nM T56556 CJ8C4Y 56951261 IC50 = 160 nM T56556 C0N9YK 57394942 IC50 = 7260 nM T56556 CTN9Q0 57396989 IC50 = 940 nM T56556 CR8MW5 57398461 IC50 = 1930 nM T56556 C9LPN4 57400130 IC50 = 3210 nM T56556 CW7B0M 57614266 IC50 = 2210 nM T56556 CQZS56 66636984 IC50 = 4100 nM T56556 C5RHD4 66637000 IC50 = 230 nM T56556 C5IT4O 70686509 IC50 = 28200 nM T56556 C9Y1TS 70686876 IC50 = 3270 nM T56556 C9B5TD 70690679 IC50 = 13300 nM T56556 CA1WO9 70696907 IC50 = 4300 nM T56556 CE1QO3 71296003 EC50 = 42 nM T56556 C2YIM8 71449571 IC50 = 5120 nM T56556 C7VGS2 71453183 IC50 = 1530 nM T56556 C1ZHB6 71453184 IC50 = 8220 nM T56556 C6ZOP0 71453185 IC50 = 970 nM T56556 CY5LI4 71454921 IC50 = 7950 nM T56556 C3OLA2 71454922 IC50 = 9350 nM T56556 C5T0NL 71454923 IC50 = 152 nM T56556 C0CIZ8 71458549 IC50 = 5910 nM T56556 CTWA64 71458550 IC50 = 5930 nM T56556 C0U5FJ 71458829 IC50 = 112 nM T56556 CA02ZE 71460396 IC50 = 3750 nM T56556 CZS0L5 71460397 IC50 = 2460 nM T56556 CPQ16X 71462088 IC50 = 6830 nM T56556 C4ZD2W 71492590 IC50 = 207 nM T56556 C0P6IG 71492759 IC50 = 176 nM T56556 C3T8ZF 71560811 EC50 = 18 nM T56556 CFN89Y 71560812 EC50 = 500 nM T56556 C42SMF 71560938 EC50 = 10000 nM T56556 C98LPJ 71560939 EC50 = 1000 nM T56556 CWCJ73 71624433 IC50 = 1100 nM T56556 CN3KI6 71624434 IC50 = 3214 nM T56556 C9RD7L 71624435 IC50 = 760 nM T56556 CGA8B3 71624544 IC50 = 544 nM T56556 C8YT2N 71624545 IC50 = 1461 nM T56556 CI7QT2 71624546 IC50 = 641 nM T56556 CA7P8Q 71624648 IC50 = 1540 nM T56556 C18BKV 71624649 IC50 = 1031 nM T56556 CMA90D 71624650 IC50 = 237 nM T56556 C3KVP8 71624651 IC50 = 591 nM T56556 CB40GR 71624766 IC50 = 943 nM T56556 CEF9J8 71624767 IC50 = 839 nM T56556 C0Z3PN 71682039 EC50 > 100000 nM T56556 CV5Z9M 71682040 EC50 > 100000 nM T56556 C1IZT7 71682041 EC50 > 100000 nM T56556 COV12T 71682195 EC50 > 100000 nM T56556 C3Y4FW 71682196 EC50 > 100000 nM T56556 CLF3I8 71682197 EC50 > 100000 nM T56556 CN6Q3L 71696716 EC50 = 12.3 nM T56556 CQCF98 71724480 EC50 = 29.5 nM T56556 C1PR7Z 71724504 EC50 = 7.2 nM T56556 CA7K8Z 71724506 EC50 = 57.5 nM T56556 CD9KH7 71724532 EC50 = 14.8 nM T56556 CWR2L5 71724556 EC50 = 0.9 nM T56556 C4ODQ2 71724557 EC50 = 160 nM T56556 C7T0UM 71724558 EC50 = 23.6 nM T56556 CUL9E2 71724582 EC50 = 38.7 nM T56556 CNW68B 71724606 EC50 = 371.7 nM T56556 CCZ9B3 71724628 EC50 = 18 nM T56556 C48CAR 72735227 IC50 = 400 nM T56556 CI6E4O 72735228 IC50 = 1550 nM T56556 CXWG13 72735229 EC50 = 3.5 nM T56556 CG7S2T 72735404 IC50 = 240 nM T56556 C2O8IJ 72735405 IC50 = 190 nM T56556 CVZK97 72735406 IC50 = 260 nM T56556 CFL45O 72735407 IC50 = 110 nM T56556 CKF0Q7 72735408 IC50 = 680 nM T56556 C5I7XA 72735580 IC50 = 610 nM T56556 CY20ED 72735581 IC50 = 470 nM T56556 C6D7QV 72735582 IC50 = 320 nM T56556 CR91NX 72735583 IC50 = 1520 nM T56556 CQ5NB6 72950792 IC50 = 426 nM T56556 CF57OZ 73346145 IC50 = 1060 nM T56556 CUX0H5 73346146 IC50 = 4270 nM T56556 C90GUQ 73347669 IC50 = 3070 nM T56556 C7KIJ0 73349189 IC50 = 2440 nM T56556 CC9F2B 73349190 IC50 = 11100 nM T56556 C7DAJ3 73352266 IC50 = 4970 nM T56556 CK3EX6 73355255 IC50 = 2710 nM T56556 CKH8D4 73355256 IC50 = 6120 nM T56556 C7NTB0 73356802 IC50 = 457 nM T56556 CIWH89 73356803 IC50 = 17900 nM T56556 C25AUR 73356804 IC50 = 4840 nM T56556 C8NC1P 76310339 EC50 = 220 nM T56556 CBDY35 76310340 EC50 = 570 nM T56556 CH9B2W 76317551 EC50 = 570 nM T56556 CVN95Y 76317552 EC50 = 530 nM T56556 C2U1VA 76321285 EC50 = 100 nM T56556 C3T5OH 76324898 EC50 = 1670 nM T56556 CCP3L1 76324899 IC50 > 2000 nM T56556 CD4V0F 76328460 IC50 = 250 nM T56556 CZ3P5R 76332141 EC50 = 80 nM T56556 C7ISD3 76335756 EC50 = 500 nM T56556 CPJ5M2 76335757 EC50 = 1270 nM T56556 CZ4SE6 76335758 EC50 = 500 nM T56556 C67ASV 76335759 EC50 = 1110 nM T56556 C5Z3GF 76335761 EC50 = 600 nM T56556 C73WDV 85922974 IC50 > 10000 nM T56556 CRB93S 89784681 EC50 = 69.3 nM T56556 CG71EX 89784708 EC50 = 28 nM T56556 C4ZOX6 89784717 EC50 = 190 nM T56556 C0ZQO6 89784722 EC50 = 32.8 nM T56556 C4U5CZ 89784733 EC50 = 54 nM T56556 CW17YB 89784735 EC50 = 59 nM T56556 C0VD4P 89784742 EC50 = 34.1 nM T56556 CZT7B9 89784751 EC50 = 47 nM T56556 CH70XJ 89784752 EC50 = 24.9 nM T56556 C6MRA2 89784753 EC50 = 24.5 nM T56556 C1JH4L 89784756 EC50 = 230 nM T56556 CN1RD8 89784760 EC50 = 195 nM T56556 C2YB6Q 89784818 EC50 = 54 nM T56556 CSK8X6 89784827 EC50 = 15.5 nM T56556 CENX80 89785043 EC50 = 32.5 nM T56556 CY46QV 89785047 EC50 = 17.5 nM T56556 CQL7T6 89785059 EC50 = 17 nM T56556 CENR59 89785064 EC50 = 235 nM T56556 CVZG56 89785117 EC50 = 86.1 nM T56556 CT43OU 89785127 EC50 = 32 nM T56556 C3FB6Q 89785132 EC50 = 30.5 nM T56556 C4S9WG 89785146 EC50 = 20 nM T56556 CCE95J 89785148 EC50 = 16.5 nM T56556 C9SBA1 89785178 EC50 = 90 nM T56556 CSI51G 89785190 EC50 = 19.7 nM T56556 CGB2P5 89785210 EC50 = 302.5 nM T56556 CTY1H5 89785238 EC50 = 48 nM T56556 CHGX10 89785254 EC50 = 195 nM T56556 CB1FR2 89794901 EC50 = 3.3 nM T56556 C43AXK 89795130 EC50 = 82.5 nM T56556 C70LJV 89795278 EC50 = 242.5 nM T56556 CFU4W2 89795305 EC50 = 152.5 nM T56556 CVB23M 89795326 EC50 = 3.6 nM T56556 CX1W9Z 89795330 EC50 = 0.9 nM T56556 C7XG4U 89795333 EC50 = 111 nM T56556 C7W1TP 89795335 EC50 = 36 nM T56556 CAX9S0 89795337 EC50 = 3.3 nM T56556 COB3Z9 89795340 EC50 = 1.7 nM T56556 C6BW0Q 89795341 EC50 = 15.8 nM T56556 COVK20 90142631 IC50 > 25000 nM T56556 CUHC90 90469229 EC50 = 3600 nM T56556 C05JQB 90469230 EC50 = 2500 nM T56556 C41EMT 90469289 EC50 = 1300 nM T56556 CA1VH0 90469291 EC50 = 2600 nM T56556 C4NX2Q 90469293 EC50 = 2600 nM T56556 C0NW8T 90469355 EC50 = 700 nM T56556 CJK73Q 90655473 EC50 = 700 nM T56556 CFX2C0 90655474 EC50 = 300 nM T56556 CYU3G9 90655475 EC50 = 400 nM T56556 CGWI98 90655476 EC50 = 15 nM T56556 C1D9TM 90655477 EC50 = 1400 nM T56556 C8A9RT 90655478 EC50 = 1100 nM T56556 CHKF72 90655479 EC50 = 2300 nM T56556 CFS75L 90655480 EC50 = 800 nM T56556 CA57QF 90655481 EC50 = 1300 nM T56556 C78PYH 90655482 EC50 = 500 nM T56556 CM1X5R 90655483 EC50 = 1100 nM T56556 CSD17I 90655484 EC50 = 1800 nM T56556 CF4Z8T 91669184 IC50 = 600 nM T56556 C3G6AI 91964346 IC50 = 953 nM T56556 CL15PA 91964352 IC50 = 300 nM T56556 C8BRG2 101876951 EC50 = 200 nM T56556 C24YLQ 101913604 IC50 = 490 nM T56556 CYM1I6 101913605 IC50 = 1600 nM T56556 CQ81YV 101913606 IC50 = 210 nM T56556 C86WSC 117777746 EC50 = 5.2 nM T56556 C9E0BT 117777811 EC50 = 4.1 nM T56556 C9YPJ7 117803128 EC50 = 25.5 nM T56556 C2UY8J 118017356 IC50 = 1700 nM T56556 CP14NL 118017358 IC50 = 1810 nM T56556 C7L8PT 118017419 IC50 = 1700 nM T56556 C7YH4G 118017423 IC50 = 610 nM T56556 C0OQ9P 118716252 EC50 = 4100 nM T56556 CK0H3V 118716255 EC50 = 400 nM T56556 C3VRT8 118716258 EC50 = 1500 nM T56556 CNS3X0 118716259 EC50 = 1300 nM T56556 CS9IV4 118716261 EC50 = 400 nM T56556 C5FD4B 118716262 EC50 = 800 nM T56556 C3BY1A 118716264 EC50 = 600 nM T56556 CLAZ45 118716265 EC50 = 3000 nM T56556 C62JPR 118716267 EC50 = 3400 nM T56556 C6JIC7 118717839 EC50 = 700 nM T56556 CLAF39 118719581 IC50 = 310 nM T56556 CHIB60 118719582 IC50 = 700 nM T56556 CFGK85 118719583 IC50 = 3000 nM T56556 CXO3V7 118719584 IC50 = 20000 nM T56556 CPI2F5 118719585 IC50 = 610 nM T56556 CCI1E7 118737162 IC50 = 184 nM T56556 C0D4GP 118737164 IC50 = 100 nM T56556 C5WYN2 118737166 IC50 = 261 nM T56556 CGT48U 118737167 IC50 = 78.9 nM T56556 CC8Q3G 118737168 IC50 = 118 nM T56556 CNZ06S 118737171 IC50 = 137 nM T56556 C3M9PE 118737173 IC50 = 451 nM T56556 C8O2WM 118737174 IC50 = 11200 nM T56556 C41ROW 118737175 IC50 = 106 nM T56556 C2UZG9 118737176 IC50 = 269 nM T56556 CUSI65 118737177 IC50 = 201 nM T56556 C85ZHJ 118737178 IC50 = 117 nM T56556 CR75MD 118737179 IC50 = 73 nM T56556 CEM28H 118737180 IC50 = 180 nM T56556 C3IH1T 118737181 IC50 = 64.2 nM T56556 C5SRA7 118737182 IC50 = 79.4 nM T56556 CU6EP1 122179376 IC50 = 357 nM T56556 CIL20J 122179390 IC50 = 45 nM T56556 C0OUW1 122179391 IC50 = 38 nM T56556 CRF71Q 122420973 IC50 = 1810 nM T56556 CCE46L 126587406 EC50 = 3.9 nM T56556 CN0LZ6 126739167 IC50 = 2330 nM T56556 CSR0Y7 127028060 IC50 > 100000 nM T56556 C8Z2XI 127028354 IC50 > 100000 nM T56556 C8Q9DG 127028355 IC50 > 100000 nM T56556 CRI72H 127028356 IC50 > 100000 nM T56556 C5A1NO 127028392 IC50 = 9640 nM T56556 CUC9I4 127040367 IC50 > 100000 nM T56556 C0I9VF 127040368 IC50 > 100000 nM T56556 CX9JE1 127040369 IC50 = 34900 nM T56556 CRM9W5 127040370 IC50 = 12000 nM T56556 CJY60W 127042304 IC50 > 100000 nM T56556 CO2P8K 127042305 IC50 = 99700 nM T56556 C56HDS 127042306 IC50 = 37600 nM T56556 CZ0E5J 127042554 IC50 = 230 nM T56556 C90ELS 127042555 IC50 = 230 nM T56556 C87PMI 127042802 IC50 = 87800 nM T56556 CRQ7U8 127042918 IC50 = 36900 nM T56556 C39PWZ 127042920 IC50 = 66600 nM T56556 C21DSU 127042921 IC50 > 100000 nM T56556 C6UZ7C 127042922 IC50 > 100000 nM T56556 CSBM31 127042943 IC50 = 12200 nM T56556 C12BJD 127042944 IC50 = 38200 nM T56556 C42ZKN 127044753 IC50 = 210 nM T56556 CA8P0B 127044754 IC50 = 310 nM T56556 CUF52K 127044901 IC50 = 840 nM T56556 CF3ML0 127044902 IC50 = 680 nM T56556 C7GXK0 127044903 IC50 = 1230 nM T56556 CP1K0B 127044904 IC50 = 390 nM T56556 CO3AX7 127044909 IC50 = 290 nM T56556 C63KNP 127044910 IC50 = 880 nM T56556 CP2U0C 127044913 IC50 = 360 nM T56556 C9SE5Y 127044914 IC50 = 3130 nM T56556 CB4JL3 127044915 IC50 = 1090 nM T56556 C9Z8XO 127045057 IC50 = 1710 nM T56556 C3FG1L 127045064 IC50 = 190 nM T56556 CM1B6D 127045208 IC50 = 1300 nM T56556 CZAL20 127045209 IC50 = 890 nM T56556 C4DH6E 127045210 IC50 = 320 nM T56556 CFX5J3 127045211 IC50 = 460 nM T56556 C5F2BE 127045212 IC50 = 970 nM T56556 CYT62M 127045213 IC50 = 680 nM T56556 C6R5MV 127045214 IC50 = 600 nM T56556 CZBJ54 127048170 IC50 = 8710 nM T56556 C6L0AF 127049502 IC50 = 8240 nM T56556 CK1SN3 127049508 IC50 = 14300 nM T56556 CB9EV4 127049509 IC50 = 6070 nM T56556 C1VP2D 127052887 IC50 = 7680 nM T56556 CG9TE5 127052888 IC50 = 9940 nM T56556 CA7N9R 127052889 IC50 = 4680 nM T56556 CX20OQ 129903920 EC50 = 10 nM T56556 CX48UI 129904103 IC50 = 1200 nM T56556 CK8S4T 132285218 IC50 = 26 nM T56556 C1WG6D 132510852 IC50 = 38 nM T56556 CH3VU5 132510853 IC50 = 29 nM T56556 C5CT0K 132547158 EC50 = 20 nM T56556 C1V7GY 134129908 IC50 = 127 nM T56556 C9VJC1 134129912 IC50 > 10000 nM T56556 CK1TS2 134129976 IC50 = 280 nM T56556 CQ5N3X 134129987 IC50 = 129 nM T56556 C3B1NJ 134130004 IC50 > 10000 nM T56556 CDG0S3 134130015 IC50 = 66.9 nM T56556 C13RTP 134130119 IC50 = 212 nM T56556 CG0NC4 134130126 IC50 = 117 nM T56556 C71PUG 134130154 IC50 = 308 nM T56556 CM40NH 134130306 IC50 > 10000 nM T56556 CCP16R 134130324 IC50 > 10000 nM T56556 C7EVF0 134130371 IC50 = 4390 nM T56556 CR6Z4W 134130497 IC50 = 150 nM T56556 C90RDH 134130514 IC50 = 223 nM T56556 CA7QF6 134130525 IC50 = 319 nM T56556 CZF1D2 134130601 IC50 = 168 nM T56556 CYLW12 134130603 IC50 > 10000 nM T56556 C63NSK 134130669 IC50 = 131 nM T56556 CK15FY 134130999 IC50 = 832 nM T56556 C6LRO0 134131064 IC50 = 208 nM T56556 C36TJZ 134131208 IC50 > 10000 nM T56556 CD69RC 134131216 IC50 = 300 nM T56556 CWP09Q 134131281 IC50 = 96.6 nM T56556 CYT40U 134131325 IC50 > 10000 nM T56556 C1JP2L 134131336 IC50 = 330 nM T56556 C6GIZ2 134131389 IC50 = 251 nM T56556 CB7A2U 134131478 IC50 = 311 nM T56556 CQ8PC9 134131521 IC50 = 679 nM T56556 C1Q0BR 134131558 IC50 = 793 nM T56556 C6QKS0 134131773 EC50 = 540 nM T56556 CDJ2L0 134133476 IC50 = 7100 nM T56556 CVRT47 134134470 IC50 = 4900 nM T56556 CA18ZH 134137512 EC50 = 4350 nM T56556 CJTO68 134140233 EC50 = 340 nM T56556 CQO05X 134141004 IC50 = 7800 nM T56556 C3PIE7 134141342 IC50 = 8900 nM T56556 CPJC31 134144364 EC50 = 380 nM T56556 C9FZI6 134147046 EC50 = 86 nM T56556 CMUK36 134147167 EC50 = 910 nM T56556 C8CIP6 134148609 EC50 = 360 nM T56556 C2Z5LD 134148627 EC50 = 360 nM T56556 CXV6P1 134149485 EC50 = 550 nM T56556 CUBF46 134149834 EC50 = 280 nM T56556 C9Q4YF 134151298 EC50 = 630 nM T56556 C48WKX 134151943 EC50 = 1050 nM T56556 CE14NO 134156590 IC50 = 7400 nM T56556 C4HTR0 134156671 EC50 = 260 nM T56556 CMN2A4 135418331 IC50 = 12800 nM T56556 C41IEM 135659059 IC50 > 20000 nM T56556 CO69BC 135885017 IC50 = 11900 nM T56556 C09BGP 135885019 IC50 = 5900 nM T56556 CV4F5D 137631464 IC50 = 507 nM T56556 COU58A 137631903 EC50 = 116 nM T56556 CL7J6T 137632165 IC50 = 128 nM T56556 CD5VI8 137632443 IC50 = 1267 nM T56556 CV09DQ 137632591 IC50 = 594 nM T56556 CXA82V 137632731 IC50 = 1100 nM T56556 C29XTR 137633043 IC50 = 621 nM T56556 CF73VM 137634351 EC50 = 85 nM T56556 CKCE38 137634438 EC50 = 72 nM T56556 C39YOJ 137634518 IC50 = 4260 nM T56556 CS26GV 137634543 IC50 = 541 nM T56556 CI2K0G 137634736 IC50 = 454 nM T56556 CB0ZJ4 137635897 EC50 = 16 nM T56556 CS3RK1 137636023 IC50 = 628 nM T56556 C54LGH 137636095 EC50 = 16 nM T56556 CI1S9R 137636359 IC50 = 146 nM T56556 C51AGO 137636525 EC50 = 8 nM T56556 CEUR16 137637400 IC50 = 605 nM T56556 CUWZ73 137637797 IC50 = 206 nM T56556 C15FLS 137638403 EC50 = 676 nM T56556 CJ57LP 137638487 EC50 = 141 nM T56556 CFL5V7 137638559 IC50 = 488 nM T56556 C1CAL5 137638992 IC50 = 882 nM T56556 CI3NO0 137639122 IC50 = 1070 nM T56556 CI5Z8K 137639498 EC50 = 47 nM T56556 CTNP09 137639885 EC50 = 4 nM T56556 C8DL5H 137639918 EC50 = 37.1 nM T56556 C5IP1S 137640378 EC50 = 210 nM T56556 C91SBQ 137640534 EC50 = 3 nM T56556 CV3QD9 137641058 EC50 = 13 nM T56556 CI0KU2 137643961 EC50 = 22 nM T56556 C36TRI 137644856 IC50 = 952 nM T56556 CS4Z5B 137644952 IC50 = 283 nM T56556 C9HCB1 137645106 EC50 = 11 nM T56556 CP42GX 137645755 IC50 = 1656 nM T56556 CN3Y8B 137646060 IC50 = 403 nM T56556 C5LFG0 137646752 EC50 = 7 nM T56556 CUP1D3 137646767 EC50 = 32 nM T56556 CTN5H3 137647282 IC50 = 2563 nM T56556 C1FM8R 137647675 EC50 = 4 nM T56556 CV2FL8 137647707 EC50 = 22 nM T56556 CVL5T7 137648146 EC50 = 79 nM T56556 CBL59T 137648334 EC50 = 8 nM T56556 CAU49L 137648335 EC50 = 4 nM T56556 C15MCA 137648533 IC50 = 838 nM T56556 CMR58G 137649090 IC50 = 164 nM T56556 C8UYC1 137649208 EC50 = 5 nM T56556 CX1NH9 137649265 EC50 = 14 nM T56556 CH07EY 137649297 IC50 = 355 nM T56556 C0W1LM 137649303 EC50 = 16 nM T56556 CYP3S6 137649349 IC50 = 325 nM T56556 CZF79C 137649780 IC50 = 1202 nM T56556 CLTE54 137650017 EC50 = 16 nM T56556 C03KMV 137650224 IC50 = 1515 nM T56556 CBAK32 137650656 IC50 = 1380 nM T56556 C5S9OL 137651096 IC50 = 512 nM T56556 C2ZVM8 137651212 IC50 = 1713 nM T56556 CC0H4S 137651220 EC50 = 82 nM T56556 C60QXZ 137651369 EC50 = 9 nM T56556 CM0SC5 137651605 EC50 = 140 nM T56556 C9PE5G 137652835 IC50 = 519 nM T56556 CDZ5I0 137652882 IC50 = 299 nM T56556 CS14NG 137652949 EC50 = 4 nM T56556 CXS2E7 137653095 EC50 = 4 nM T56556 C2B9JN 137653194 IC50 = 472 nM T56556 CN6QH5 137653329 EC50 = 85 nM T56556 C65IAD 137653455 IC50 = 985 nM T56556 C59ZRO 137653532 IC50 = 910 nM T56556 CB1Y8V 137655046 IC50 = 348 nM T56556 C6RP1Z 137655517 IC50 = 354 nM T56556 C89NMB 137655783 IC50 = 1530 nM T56556 C12YJV 137655818 IC50 = 5270 nM T56556 CTV4I1 137655973 IC50 = 122 nM T56556 C0N1TD 137656929 IC50 = 866 nM T56556 COY89M 137657641 EC50 = 145 nM T56556 C5C0KF 137658808 EC50 = 1540 nM T56556 CTO85K 137659047 IC50 = 6400 nM T56556 CB8CJ2 137659409 IC50 = 691 nM T56556 C9HU7R 137659989 IC50 = 325 nM T56556 C8MXN5 137661038 EC50 = 2 nM T56556 C31GEP 137661880 IC50 = 750 nM T56556 CPI3E4 137662036 IC50 = 1630 nM T56556 C7SH6Z 137662093 EC50 = 12 nM T56556 CP1M2F 137662213 IC50 = 2121 nM T56556 CC1QL5 139593871 IC50 = 2130 nM T56556 C5PKZ2 139593897 IC50 = 951 nM T56556 C9USZ1 145949183 EC50 = 4 nM T56556 C3H7QO 145949352 EC50 = 29 nM T56556 C43QGK 145949445 IC50 = 284 nM T56556 CFN6T2 145949660 EC50 = 11 nM T56556 C2X7WS 145950031 IC50 = 44.8 nM T56556 CHB1S3 145950435 IC50 = 57.7 nM T56556 CZRP27 145950520 IC50 = 51.5 nM T56556 CB7KD0 145950545 EC50 = 2 nM T56556 CUB64Y 145950625 EC50 = 690 nM T56556 CNG6V3 145950683 IC50 = 78.7 nM T56556 CK6YR0 145950764 EC50 = 19.5 nM T56556 C07XUY 145950844 IC50 = 61.4 nM T56556 C94HRD 145950874 EC50 = 577 nM T56556 CE4SY2 145950964 IC50 = 1150 nM T56556 CUY09I 145950988 IC50 = 127 nM T56556 CIZ82R 145951128 IC50 = 1040 nM T56556 CR31OX 145951139 IC50 = 336 nM T56556 C4TRJ3 145951213 IC50 = 799 nM T56556 C53MCJ 145951316 IC50 = 65.3 nM T56556 CSYV28 145951611 EC50 = 19 nM T56556 CUD94F 145952004 EC50 = 63 nM T56556 C8Y7ND 145952143 IC50 = 66.3 nM T56556 C5V1MZ 145952691 IC50 = 801 nM T56556 C9O3IC 145952963 IC50 = 1770 nM T56556 C1L4NV 145953000 EC50 = 0.6 nM T56556 CIF74V 145953301 IC50 = 726 nM T56556 C5Z0BT 145953360 IC50 = 33 nM T56556 COSR30 145953465 IC50 = 369 nM T56556 CW97IA 145953788 IC50 = 904 nM T56556 CC3GQ9 145954340 EC50 = 21.8 nM T56556 C21XAV 145954560 EC50 = 1230 nM T56556 C2KBR1 145954586 IC50 = 30.2 nM T56556 CQ7Y6U 145955013 EC50 = 48 nM T56556 C7LP2U 145955206 EC50 = 6 nM T56556 CJ3ET0 145955421 EC50 = 10 nM T56556 CBI96G 145955592 IC50 = 20 nM T56556 C06LAX 145955721 IC50 = 2120 nM T56556 C3CAG9 145955791 IC50 = 221 nM T56556 CM62WT 145956236 IC50 = 120 nM T56556 CHCB46 145956407 EC50 = 4 nM T56556 C6FS8J 145956778 IC50 = 119 nM T56556 CLD32M 145957548 IC50 = 48.2 nM T56556 C8ZAT2 145957575 IC50 = 44.8 nM T56556 CX32LO 145957840 IC50 = 106 nM T56556 C9F8TW 145957857 EC50 = 48.3 nM T56556 CXH7F4 145957934 IC50 = 820 nM T56556 CB5PZ6 145958054 EC50 = 71.2 nM T56556 CB9CF1 145958160 EC50 = 14 nM T56556 CL15OJ 145958265 EC50 = 10 nM T56556 C9QO8G 145958364 IC50 = 16200 nM T56556 CL76TP 145958566 IC50 = 1190 nM T56556 CDH0A1 145958606 IC50 = 642 nM T56556 CD46YZ 145958660 IC50 = 1640 nM T56556 C0T5ZE 145958944 IC50 = 1620 nM T56556 CBQ8K0 145959274 IC50 = 795 nM T56556 CPU4D2 145959408 IC50 = 33.1 nM T56556 C3ZLR8 145959442 IC50 = 84 nM T56556 C2XSC1 145959549 IC50 = 49.1 nM T56556 C4PQ5A 145959673 IC50 = 811 nM T56556 C3C6SA 145959746 EC50 = 34 nM T56556 CIA08G 145959888 IC50 = 101 nM T56556 CVX17O 145960171 EC50 = 5 nM T56556 CYL21E 145960198 IC50 = 570 nM T56556 C2T8PH 145960322 IC50 = 610 nM T56556 CR0J2I 145960997 IC50 = 57.2 nM T56556 CA7RL9 145962283 IC50 = 5310 nM T56556 CBU79J 145964049 IC50 = 501 nM T56556 C1A7DH 145964067 IC50 = 9930 nM T56556 C5YP9J 145964072 IC50 = 6910 nM T56556 C80ESB 145964513 IC50 = 1060 nM T56556 CM5W0B 145964551 IC50 = 733 nM T56556 CNM1G3 145964790 IC50 = 766 nM T56556 C2QI8W 145965708 IC50 = 90 nM T56556 CJRZ24 145966467 IC50 = 445 nM T56556 C4OZH5 145966511 IC50 = 880 nM T56556 CBL6O0 145966757 IC50 = 7670 nM T56556 C4ZA8I 145966835 IC50 = 1550 nM T56556 CVB80Y 145966874 IC50 = 14390 nM T56556 C58UJF 145968465 IC50 = 15800 nM T56556 CTP6I7 145971735 IC50 = 646 nM T56556 CYU1W6 145971955 EC50 = 11 nM T56556 CZ3N8M 145972213 IC50 = 210 nM T56556 CIT6S0 145972309 IC50 = 18500 nM T56556 C6DKL1 145972800 IC50 = 438 nM T56556 C9QW5V 145973127 IC50 = 59 nM T56556 C96ARL 145973335 IC50 = 3230 nM T56556 C65PUC 145973732 IC50 = 6730 nM T56556 CM1UP7 145973867 IC50 = 430 nM T56556 C14UYO 145974134 IC50 = 287 nM T56556 C8K3YC 145974263 IC50 = 130 nM T56556 C1CKI3 145974543 IC50 = 297 nM T56556 CH30BM 145974617 IC50 = 270 nM T56556 CGWT84 145974788 EC50 = 4 nM T56556 C2O0FG 145974893 IC50 = 351 nM T56556 CLZ4D7 145974899 IC50 = 8760 nM T56556 CQ53WA 145974921 IC50 = 1400 nM T56556 CZ4I8A 145975509 IC50 = 61.6 nM T56556 CAF5H4 145975609 IC50 = 9000 nM T56556 CRO97S 145975756 IC50 = 2830 nM T56556 CM05IS 145975969 IC50 = 176 nM T56556 CA3V5K 145976004 IC50 = 15300 nM T56556 CT4C0Y 145976071 IC50 = 23240 nM T56556 C3PU1W 145976134 IC50 = 77.4 nM T56556 CM0DC2 145976272 IC50 = 2720 nM T56556 CZ9EA3 145976337 IC50 = 4080 nM T56556 C7EP8H 145976472 IC50 = 6650 nM T56556 CV9W1U 145976531 IC50 = 39800 nM T56556 COA43R 145976548 IC50 = 190 nM T56556 C6SV1M 145976742 IC50 = 11400 nM T56556 C6W1PJ 145977012 IC50 = 228 nM T56556 CZP74I 145977357 IC50 = 129 nM T56556 CQ6PN4 145977383 IC50 = 8340 nM T56556 CB7WX4 145977891 IC50 = 102 nM T56556 CK89HF 145978336 IC50 = 2130 nM T56556 C3Q8JT 145978355 IC50 = 1130 nM T56556 C53TFX 145978471 IC50 = 259 nM T56556 C4S5RJ 145978614 IC50 = 287 nM T56556 C3FSQ9 145978662 IC50 = 267 nM T56556 CGY0D8 145978682 IC50 = 2360 nM T56556 CL4WJ5 145978764 IC50 = 565 nM T56556 CF8L7A 145979103 EC50 = 22.3 nM T56556 CM6Z4G 145979318 EC50 = 989 nM T56556 CDYJ89 145979389 IC50 = 5400 nM T56556 C3EX7W 145979504 EC50 = 51.7 nM T56556 C24OSG 145979776 IC50 = 8440 nM T56556 C4G7LT 145980033 EC50 = 38.3 nM T56556 CUSP05 145981621 IC50 = 10900 nM T56556 C26OWY 145981942 EC50 = 19.9 nM T56556 C10YDI 145982128 EC50 = 1170 nM T56556 CZ9N5Q 145982445 IC50 = 6950 nM T56556 C3ZG6V 145982714 IC50 = 6630 nM T56556 C13VFZ 145985646 EC50 = 6.4 nM T56556 CU1Z8M 145986566 EC50 = 1390 nM T56556 C37ULP 145986567 IC50 = 10000 nM T56556 C3KFN7 145987093 EC50 = 448 nM T56556 CFU24J 145987833 EC50 = 3.1 nM T56556 CGL02K 145988126 EC50 = 57 nM T56556 C4F5OW 145988257 IC50 = 20100 nM T56556 CCIF35 145989307 IC50 = 12000 nM T56556 CX3YR7 145990226 EC50 = 34.7 nM T56556 CN1V8K 145992500 EC50 = 7.4 nM T56556 CT02XU 145992768 EC50 = 14 nM T56556 CKZA78 145992770 EC50 = 107 nM T56556 C07OTB 145993028 EC50 = 25.2 nM T56556 C65JUT 145993130 EC50 = 10.9 nM T56556 C8WF7P 145993760 IC50 = 6330 nM T56556 C3UC5J 145994097 EC50 = 59.7 nM T56556 CKM79V 145994277 EC50 = 27.1 nM T56556 CF92IR 155510784 EC50 > 100000 nM T56556 C3MZ1E 155511724 EC50 = 2300 nM T56556 CE4C1X 155512695 IC50 = 1630 nM T56556 CC9X1U 155514114 IC50 = 13100 nM T56556 CVZ7D2 155514151 EC50 = 4600 nM T56556 C0AFT8 155514623 EC50 = 2.4 nM T56556 C17AZU 155515244 EC50 = 5100 nM T56556 CUHI07 155515592 IC50 = 994 nM T56556 CH6O3X 155515825 EC50 = 16000 nM T56556 CV9TF6 155516191 EC50 = 2.2 nM T56556 C75VID 155517095 EC50 = 46 nM T56556 C4IS7E 155518051 EC50 = 4500 nM T56556 CLQO05 155518383 IC50 = 202 nM T56556 CCL04Y 155518581 IC50 = 7400 nM T56556 CCK94U 155519382 IC50 = 2570 nM T56556 CA1BD2 155520579 EC50 = 3700 nM T56556 CE50TP 155521906 IC50 = 7270 nM T56556 C97CDW 155522930 IC50 = 20000 nM T56556 CS18PU 155523410 EC50 = 33500 nM T56556 CN6ST7 155523417 EC50 = 1.1 nM T56556 C1V9YM 155523822 EC50 = 3000 nM T56556 CBZ8K4 155524289 IC50 = 513 nM T56556 C4LK0P 155524329 IC50 = 47.3 nM T56556 C86ZPR 155525910 EC50 = 8100 nM T56556 C8C7VA 155525927 EC50 > 100000 nM T56556 C8TQ4G 155526547 EC50 = 13.5 nM T56556 C7WI3R 155526594 IC50 = 1070 nM T56556 CTW8I2 155526857 EC50 = 3800 nM T56556 C41JTR 155528166 EC50 = 5600 nM T56556 C9BGT5 155528240 EC50 = 55.4 nM T56556 C75OQS 155529248 IC50 = 1900 nM T56556 C56AHP 155530068 EC50 = 3.5 nM T56556 CE0F4W 155530435 IC50 = 3669 nM T56556 C2PW4J 155530538 IC50 = 2025 nM T56556 CQZD59 155530897 IC50 = 3948 nM T56556 C1HFX4 155531129 EC50 = 7200 nM T56556 CUL2G4 155531672 EC50 > 1000 nM T56556 C4IW9M 155533366 EC50 = 41000 nM T56556 C9QT4A 155533532 IC50 = 7.98 nM T56556 CRC20Y 155534149 EC50 = 6400 nM T56556 CP9C0M 155534240 EC50 = 1220 nM T56556 C52RYM 155534490 IC50 = 178 nM T56556 CHF7A6 155535686 EC50 = 84 nM T56556 COFC46 155536723 EC50 = 4700 nM T56556 CP3U4C 155536912 EC50 = 46000 nM T56556 CYG84N 155537154 EC50 = 9500 nM T56556 CB1FI9 155537197 EC50 = 793 nM T56556 C2J7TM 155537461 IC50 = 652 nM T56556 CGD47O 155537584 EC50 = 2.1 nM T56556 C8FX4B 155537647 IC50 = 5650 nM T56556 CVES34 155538494 EC50 = 2300 nM T56556 CS4WO9 155538718 IC50 = 10500 nM T56556 CFN41J 155538958 EC50 = 6200 nM T56556 C8WT1F 155539055 IC50 = 1460 nM T56556 CLU37N 155539307 EC50 = 8100 nM T56556 C9VW3C 155539729 IC50 = 31 nM T56556 C70PUH 155540561 IC50 = 335 nM T56556 CL9G5X 155541828 IC50 > 10000 nM T56556 CE0G9A 155542384 IC50 = 1100 nM T56556 C56DUX 155543049 IC50 > 10000 nM T56556 CP93FH 155543149 EC50 = 6800 nM T56556 CJ5Q2K 155543420 IC50 = 10080 nM T56556 C7JUC3 155543680 EC50 = 3800 nM T56556 CYE3M6 155544628 IC50 = 556 nM T56556 C0GVI7 155545772 EC50 = 1800 nM T56556 CQ3S7A 155545818 IC50 > 10000 nM T56556 CMIN20 155545978 IC50 = 846 nM T56556 CDO86V 155546844 IC50 = 1780 nM T56556 CEA2R7 155547184 IC50 = 2900 nM T56556 COM08I 155547388 IC50 = 1320 nM T56556 CDY82R 155549328 EC50 = 4600 nM T56556 C86HEA 155549333 IC50 = 811 nM T56556 C72IFK 155549366 IC50 = 10400 nM T56556 CDFC58 155549450 IC50 = 1230 nM T56556 C53PGC 155550195 EC50 = 446 nM T56556 CWK3L0 155550287 EC50 = 11000 nM T56556 CB8FC1 155550293 EC50 = 4300 nM T56556 C8F3HQ 155550402 IC50 = 2000 nM T56556 CGF1W0 155551433 IC50 = 1920 nM T56556 CP7A5R 155552128 EC50 = 3900 nM T56556 CIF4T8 155553306 EC50 = 2.8 nM T56556 CG9K4Y 155553476 EC50 > 100000 nM T56556 C5QE9O 155553583 IC50 = 1030 nM T56556 CEZ7B1 155554618 EC50 = 6.5 nM T56556 CX6CM0 155554919 EC50 = 64 nM T56556 C2Y9UG 155554959 EC50 = 2300 nM T56556 C7JI4C 155555932 EC50 = 60 nM T56556 C8M0BP 155556108 IC50 = 989 nM T56556 CDAP41 155557648 IC50 = 202 nM T56556 CG0H8N 155557744 EC50 = 3300 nM T56556 CM2J5L 155558116 EC50 = 6400 nM T56556 C27XQN 155558615 EC50 = 7.2 nM T56556 CUNV65 155558919 EC50 = 17.8 nM T56556 C21LPY 155559292 IC50 = 1260 nM T56556 CG6NC7 155560071 EC50 = 4200 nM T56556 C46KOL 155560381 IC50 = 698 nM T56556 CY6UB5 155561091 IC50 = 112 nM T56556 CS2B6P 155561257 EC50 = 97 nM T56556 C6VUX2 155561896 IC50 = 77.3 nM T56556 CX42YD 155562157 IC50 > 10000 nM T56556 CPOI59 155562875 IC50 = 883 nM T56556 CWM67C 155563340 EC50 = 2500 nM T56556 CS0NC2 155563858 IC50 = 805 nM T56556 CJ57SV 155563869 IC50 > 10000 nM T56556 CU1TG6 155564277 IC50 = 7820 nM T56556 CJ4GX0 155564603 IC50 = 1060 nM T56556 C7SMU4 155565022 IC50 = 1100 nM T56556 C6Z2XK 155566234 EC50 = 4700 nM T56556 CAN76P 155566986 EC50 > 100000 nM T56556 C8ZE6S 155567126 IC50 = 4490 nM T56556 CO1LU7 155567143 EC50 = 30.7 nM T56556 C9QA2H 155567258 IC50 = 4780 nM T56556 CHT79A 155568041 EC50 = 5900 nM T56556 CFCV37 155568122 IC50 = 14800 nM T56556 CTV5K3 155568177 EC50 = 24.5 nM T56556 C03SJY 155568508 EC50 = 2 nM T56556 CO08ZV 155568670 EC50 = 5400 nM T56556 CTXV81 155568869 EC50 = 2.4 nM T56556 COQJ76 155569267 IC50 = 1450 nM T56556 D00RIX 5280443 IC50 = 3100 nM T56556 D01UYI 5281607 IC50 = 1500 nM T56556 D02ZRO 735125 IC50 = 1080 nM T56556 D04GYT 15511439 IC50 = 3981.07 nM T56556 D07RSH 631105 IC50 = 5980 nM T56556 D09HIM 22004473 IC50 = 3890.45 nM T56556 D0A4TF 15511440 IC50 = 5011.87 nM T56556 D0E5IP 3795 EC50 = 189 nM T56556 D0G3TK 5280863 IC50 = 4700 nM T56556 D0I7GE 11790 IC50 = 1310 nM T56556 D0NJ4H 5281670 IC50 = 49000 nM T56556 D0S0RK 10680 IC50 = 17000 nM T56556 D0S8CE 15950351 IC50 = 676.08 nM T75907 C79IRE 71620755 IC50 = 360 nM T75907 C7PI9C 71620756 IC50 = 360 nM T75907 CGD70V 71620759 IC50 = 360 nM T75907 CX85HD 71621073 IC50 = 360 nM T75907 CZB46R 71621227 IC50 = 360 nM T75907 CNP1U5 86574151 IC50 = 360 nM T75907 C2LM9W 127026354 IC50 = 30 nM T75907 CRD02W 127026355 IC50 = 280 nM T75907 C6KE3B 127026667 IC50 = 80 nM T75907 CE2PX6 127026668 IC50 = 30 nM T75907 C7VP6A 127026669 IC50 = 10 nM T75907 C1IF8B 127028921 IC50 = 70 nM T75907 C5ZK6J 127029217 IC50 = 50 nM T75907 CZ3DS8 127029218 IC50 = 40 nM T75907 CMR68I 127029233 IC50 = 1 nM T75907 C7ZHE4 127029234 IC50 = 10 nM T75440 D01XOD 54897 Ki = 0.5 nM T75440 D04BNP 5391 IC50 = 62517269.28 nM T75440 D07JVL 3016 IC50 = 123594743.3 nM T75440 D09LDR 4616 IC50 = 55590425.73 nM T75440 D0CP4E 2802 IC50 = 555904257.3 nM T75440 D0E0OG 3958 IC50 = 285759054.3 nM T75440 D0T5WK 4506 IC50 = 100000000 nM T75440 D0W2NM 3380 IC50 = 263026799.2 nM T75440 D0Z5OV 17925 IC50 = 555904257.3 nM T75440 D0Z9VB 31640 IC50 = 10864256.24 nM T75440 D0G4YZ 11653141 Ki = 2.47 nM T75440 D0M2TS 71600087 IC50 = 800 nM T75440 D01LOJ 11595759 Ki = 6.68 nM T75440 D0FR9I 10430788 Ki = 0.188 nM T75440 D0ZK2Q 9841240 Ki = 2.5 nM T75440 D05UXF 6433109 Ki = 6.4 nM T75440 D08AWI 11430856 Ki > 2000 nM T75440 D0K5IQ 9844410 IC50 = 0.92 nM T75440 D0VN4K 1345 IC50 = 1.1 nM T75440 CCH08A 2997 IC50 = 106414301.8 nM T75440 C87SBM 4540 IC50 = 500034535 nM T75440 CWB1Y9 15024 IC50 = 285759054.3 nM T75440 C2B9SE 16795 IC50 = 76913044.03 nM T75440 CC9L3A 19011 IC50 = 2630267.99 nM T75440 CHL67Q 30401 IC50 = 40831938.63 nM T75440 C7H2PJ 65764 IC50 = 2328091.26 nM T75440 CSTD39 75849 IC50 = 25003453.62 nM T75440 CL25FN 76175 IC50 = 2857590.54 nM T75440 CV8O9T 78641 IC50 = 2588212.92 nM T75440 CB0PY6 92294 IC50 = 15381546.4 nM T75440 CJD8Z6 118749 IC50 = 345143739.3 nM T75440 CYOL58 128744 IC50 = 142889395.9 nM T75440 CH2JA9 148760 IC50 = 10423174.29 nM T75440 CIUV59 188298 IC50 = 13335214.32 nM T75440 C1RK6L 520217 IC50 = 666806769.2 nM T75440 CNA35U 528222 IC50 = 454988060.2 nM T75440 CQ8H2P 622885 IC50 = 1614358.56 nM T75440 C89UHQ 5458184 Ki = 0.242 nM T75440 C01SQJ 6603782 Ki = 0.41 nM T75440 CR5NV7 9975396 IC50 = 181970085.9 nM T75440 C48VJA 10264786 IC50 = 27797132.68 nM T75440 CM8L2J 10358803 IC50 = 277971326.8 nM T75440 C8MT4I 10453776 Ki = 3.9 nM T75440 C3QEM9 10469149 IC50 = 263026799.2 nM T75440 CYX7O2 10738832 Ki = 1.6 nM T75440 CR67IU 10833643 IC50 = 11.8 nM T75440 CFJG64 11059058 IC50 = 1040 nM T75440 CR97ZW 11488150 Ki = 2.68 nM T75440 CR6OL3 11780929 Ki = 30.1 nM T75440 CXLW54 11948707 Ki > 10000 nM T75440 CM1T4V 12790028 IC50 = 142889395.9 nM T75440 C50BWX 13292074 IC50 = 47643098.68 nM T75440 CLH94F 13485706 IC50 = 416869383.5 nM T75440 CKZI28 15294055 IC50 = 620 nM T75440 CZ2IS9 16660294 Ki > 10000 nM T75440 C3W8DT 16749353 IC50 > 5000 nM T75440 CCP1J0 20542073 IC50 = 33342641.28 nM T75440 CDJ23A 23275339 IC50 = 2172701.18 nM T75440 CSB68Q 23275675 IC50 = 195884467.4 nM T75440 CWYX46 23275762 IC50 = 35727283.82 nM T75440 C9S0VL 23275763 IC50 = 625172692.8 nM T75440 CHL6M4 23275854 IC50 = 55590425.73 nM T75440 CTG41H 24778289 IC50 > 2000 nM T75440 C54TYJ 24945827 Ki = 0.882 nM T75440 CL6RD3 25140330 Ki = 0.537 nM T75440 CV4ZB3 25140479 Ki = 0.15 nM T75440 CD5V1U 25140760 Ki = 0.86 nM T75440 CIKB38 25208880 Ki = 0.997 nM T75440 C0RWI9 44366034 IC50 = 23280912.58 nM T75440 CFG7O1 44366036 IC50 = 41686938.35 nM T75440 CF72JC 44366089 IC50 = 25003453.62 nM T75440 CG9YJ7 44366116 IC50 = 135207256.3 nM T75440 CQ19LG 44366138 IC50 = 71449632.61 nM T75440 C1X5TW 44366161 IC50 = 188799134.9 nM T75440 C4LPC1 44366162 IC50 = 20417379.45 nM T75440 C8LT0S 44366169 IC50 = 52601726.64 nM T75440 C24VAZ 44366175 IC50 = 3334264.13 nM T75440 C26GHA 44366179 IC50 = 58884365.54 nM T75440 CR2V5W 44366192 IC50 = 833681184.6 nM T75440 CNAU14 44366206 IC50 = 285759054.3 nM T75440 CL7MP2 44366219 IC50 = 333426412.8 nM T75440 C94OVZ 44366228 IC50 = 188799134.9 nM T75440 CSF51U 44366236 IC50 = 243781081.8 nM T75440 CIP40L 44366255 IC50 = 52601726.64 nM T75440 C5TOJ7 46853447 IC50 = 2000 nM T75440 C8ZCU1 50994211 Ki = 1.57 nM T75440 CMJ62D 53245590 Ki = 2540 nM T75440 C49IKC 56671767 Ki = 1.19 nM T75440 C9D8WH 68968012 IC50 = 1.6 nM T75440 C1U2OK 72793912 Ki = 8 nM T75440 C0ZT5N 90644973 Ki = 293 nM T75440 CWE5X6 90656115 IC50 = 350 nM T75440 CLM5N2 90656116 IC50 = 680 nM T75440 CEAH51 118731302 Ki = 0.87 nM T75440 C5X8MN 122186880 Ki = 2897 nM T75440 C7ODW3 122195524 Ki > 900 nM T75440 CEK04Y 122196423 Ki = 28.13 nM T75440 C7ZKE3 122196424 Ki = 224.46 nM T75440 CVLH25 122196425 Ki = 29.11 nM T75440 C2HUV5 122196426 Ki > 10000 nM T75440 C5L9BD 134143752 Ki = 2100 nM T75440 C71PIY 134144970 Ki = 2200 nM T75440 CGS61F 137553161 Ki = 2930 nM T75440 CD7X5J 145951649 Ki = 28.9 nM T75440 CI4F0U 145954243 Ki = 25.4 nM T75440 CUSI97 145954858 Ki = 54.3 nM T75440 CKA9Z4 145958209 Ki = 70 nM T75440 C9ZY4V 145960315 Ki = 31.5 nM T75440 CPN90L 145971987 Ki = 31.6 nM T75440 CCTO46 155512230 Ki > 10000 nM T75440 CV35ZN 155513505 Ki = 3980 nM T75440 CB65EC 155513663 Ki = 96.1 nM T75440 C23PQH 155514371 Ki = 243 nM T75440 CLD73A 155514689 Ki = 1531.3 nM T75440 CWH24L 155517967 Ki = 562.5 nM T75440 CB0JS3 155518392 Ki > 10000 nM T75440 CH4ZC6 155518977 Ki = 53 nM T75440 C8DNZ6 155519967 Ki = 4737.3 nM T75440 CKH8G2 155522433 Ki > 10000 nM T75440 C36DYH 155525138 IC50 = 2.13 nM T75440 CIW07A 155526405 Ki = 3.2 nM T75440 C2UL4X 155526804 Ki > 10000 nM T75440 C1O0IC 155527848 Ki > 10000 nM T75440 C78XNA 155528306 Ki = 385.3 nM T75440 C2XY8U 155531728 Ki = 184.2 nM T75440 CY0H3U 155533272 Ki = 2020 nM T75440 COT9U8 155535203 Ki = 2380 nM T75440 CTD7J5 155537862 Ki = 462.3 nM T75440 C4C9NY 155541492 Ki > 10000 nM T75440 C1LU5B 155541865 Ki = 200 nM T75440 CMT60C 155543832 Ki = 2890 nM T75440 CJS87Q 155545399 Ki = 3170 nM T75440 C1L0SN 155547768 Ki = 200.7 nM T75440 CJ61KL 155547788 Ki = 369 nM T75440 CRY61B 155548339 Ki = 1696 nM T75440 C6IL4E 155548476 Ki = 50 nM T75440 CGL97X 155555425 Ki > 10000 nM T75440 CDL16X 155555765 Ki = 693.8 nM T75440 CBS89O 155556618 Ki = 2020 nM T75440 CLQH75 155558424 Ki = 208.4 nM T75440 CIPF89 155559210 Ki = 214 nM T75440 CAQ4S5 155561301 Ki > 10000 nM T75440 CCOD50 155562467 Ki = 2220 nM T75440 COP4K5 155562523 Ki > 10000 nM T75440 CI12LD 155566336 Ki > 10000 nM T75440 CU9HA1 155566889 Ki > 10000 nM T75440 C13REG 44471685 Ki = 3166 nM T75440 C6VJE1 6603767 Ki = 4.5 nM T75440 C9TZG6 9842567 Ki = 1.4 nM T75440 D06DTT 193319 IC50 = 71449632.61 nM T75440 D0A0ED 132496 Ki = 3.25 nM T75440 D0FF6S 16038374 IC50 > 2000 nM T75440 D0O6JQ 24839733 Ki = 13.6 nM T94621 D03ZBT 11626560 IC50 > 10000 nM T94621 D01NEC 51042438 IC50 = 1 nM T94621 D01ZAQ 25227436 IC50 = 8 nM T94621 D02ZQS 16095342 IC50 = 1350 nM T94621 D09IYM 24905401 IC50 = 402 nM T94621 D0E3TC 44259 IC50 = 6.5 nM T94621 D0I4TH 24788740 IC50 = 18 nM T94621 D0MS3Z 16725726 Ki = 4 nM T94621 D0W3RW 24964624 IC50 = 12 nM T94621 D03BNU 59604787 IC50 > 10000 nM T94621 D0ZE5U 11161844 IC50 = 5 nM T94621 D0T3ME 156422 IC50 > 30000 nM T94621 COYW98 9222 IC50 > 100000 nM T94621 C3XD4Z 139106 IC50 = 135000 nM T94621 C5EH9L 139601 IC50 = 80000 nM T94621 CU73ST 599501 IC50 = 660000 nM T94621 CFC7G1 756695 IC50 = 41000 nM T94621 C1SVD2 2132479 IC50 = 1900 nM T94621 C9ZT2G 2753118 IC50 = 72000 nM T94621 CFY1D0 2974957 IC50 > 10000 nM T94621 CABJ52 3129049 IC50 = 59000 nM T94621 C98ITU 5327109 IC50 = 260 nM T94621 CWN6P7 5702541 IC50 = 590 nM T94621 CG17TN 6914611 IC50 = 6.8 nM T94621 C7E2QK 6914613 IC50 = 257 nM T94621 CIAL53 9819282 IC50 = 23000 nM T94621 CC7Y2O 9828163 IC50 = 220 nM T94621 C8QZD6 9829528 IC50 = 26 nM T94621 C16VXB 9863538 IC50 > 10000 nM T94621 CI0AW6 9871034 IC50 = 2057 nM T94621 C7H8EO 9871171 IC50 = 7356 nM T94621 C18HKQ 9885748 IC50 = 720 nM T94621 CUE4B5 9912061 IC50 > 50000 nM T94621 CU7FH2 9957031 IC50 > 50000 nM T94621 CJX43Z 10055074 IC50 = 359 nM T94621 CEV18B 10128689 IC50 > 50000 nM T94621 C7PK4U 10152003 IC50 = 15700 nM T94621 C4FUG5 10152760 IC50 = 4517 nM T94621 CMO32F 10152761 IC50 = 325 nM T94621 CMR17F 10174144 IC50 > 50000 nM T94621 CLP79V 10196532 IC50 = 388 nM T94621 CI8MW4 10216627 IC50 = 5 nM T94621 C0O8FI 10217663 IC50 = 1179 nM T94621 CY6MJ3 10218178 Ki = 325 nM T94621 CT97JL 10218280 IC50 = 577 nM T94621 C8V6RI 10240275 IC50 = 212 nM T94621 CD3W6Y 10289038 IC50 > 20000 nM T94621 C2LP9A 10289671 IC50 = 300 nM T94621 CT0M7Q 10311653 IC50 = 259 nM T94621 C4MOF8 10312133 IC50 = 144 nM T94621 CAK9U4 10415819 IC50 = 65 nM T94621 CNY45Z 11151075 IC50 = 10 nM T94621 CO48BE 11165629 IC50 = 14 nM T94621 CO2DA6 11165945 IC50 = 10 nM T94621 C53MZX 11168481 IC50 > 50000 nM T94621 C1GYU5 11175137 IC50 = 18000 nM T94621 C3IJ6D 11180030 IC50 > 50000 nM T94621 CPVK21 11180486 IC50 = 1228 nM T94621 CMA1U5 11196322 IC50 = 510 nM T94621 C7BN5E 11225451 IC50 > 50000 nM T94621 CC6V3Z 11225497 IC50 = 529 nM T94621 C1UZC6 11226082 IC50 = 37720 nM T94621 CKB72H 11237628 IC50 = 8141 nM T94621 CL0QN6 11246027 IC50 = 27 nM T94621 C2ON6C 11246455 IC50 = 118 nM T94621 CCF0G6 11249067 IC50 = 2062 nM T94621 C49NET 11256399 IC50 = 204 nM T94621 C3T6XF 11256709 IC50 = 8 nM T94621 C1TCF3 11260243 IC50 > 50000 nM T94621 COHW29 11272514 IC50 > 50000 nM T94621 C9FG0K 11293497 IC50 = 4 nM T94621 CBOP58 11293798 Ki = 1120 nM T94621 CHBC32 11296432 IC50 = 839 nM T94621 CO39LB 11312547 IC50 = 31000 nM T94621 C1KOA4 11325683 IC50 = 39 nM T94621 CPV82H 11341558 IC50 > 50000 nM T94621 C26BZX 11362471 Ki = 3970 nM T94621 C4G3RZ 11364261 IC50 > 50000 nM T94621 COF6V0 11370369 IC50 = 9 nM T94621 C5EP3S 11373564 IC50 = 11 nM T94621 C1LT9H 11374804 IC50 > 50000 nM T94621 CD2P0L 11383042 IC50 = 5 nM T94621 CWXB93 11397177 Ki > 10000 nM T94621 CPFW90 11399527 IC50 = 556 nM T94621 CRC7H2 11407608 IC50 = 29 nM T94621 C6KQ2U 11409661 IC50 > 50000 nM T94621 C4L5TF 11409804 IC50 = 7356 nM T94621 C4OT0X 11417334 IC50 = 10 nM T94621 CCP18F 11430140 IC50 = 6 nM T94621 C1FC5U 11431759 IC50 > 50000 nM T94621 CW53GT 11440050 IC50 = 57 nM T94621 C5H7KT 11453730 IC50 = 3 nM T94621 CI9L2T 11454186 IC50 > 50000 nM T94621 CQS3U5 11454871 IC50 > 50000 nM T94621 CE72WO 11489421 IC50 = 15390 nM T94621 C7XM4C 11504922 IC50 = 59 nM T94621 CPN02A 11513279 IC50 = 27 nM T94621 C38OKZ 11513374 IC50 = 177 nM T94621 C85JUO 11514232 IC50 = 1600 nM T94621 CJ7XT8 11526364 IC50 = 1909 nM T94621 CTM2Q3 11526695 IC50 = 85 nM T94621 CEX8Y5 11527102 IC50 = 44 nM T94621 C5NPU9 11534762 IC50 = 5127 nM T94621 CCJ7Z1 11535873 IC50 = 830 nM T94621 CTG83F 11539329 Ki > 8400 nM T94621 CG84SZ 11540975 IC50 = 1572 nM T94621 CWCN15 11541348 IC50 = 44 nM T94621 CY0JX9 11541985 IC50 = 21 nM T94621 CSCJ29 11542208 IC50 = 229 nM T94621 C2O3DZ 11543058 IC50 = 880 nM T94621 CA8R0K 11547290 IC50 = 928 nM T94621 CX96EC 11549174 IC50 = 22 nM T94621 C3Z8PI 11549180 IC50 = 31 nM T94621 CJEB45 11549190 IC50 = 2106 nM T94621 CJF21M 11549537 IC50 = 297 nM T94621 CN25UD 11556452 IC50 = 99 nM T94621 CACS26 11561968 Ki > 10000 nM T94621 C3WVM7 11564772 IC50 = 180 nM T94621 C4LI8C 11564882 IC50 = 770 nM T94621 C9LDN1 11577612 IC50 = 107.2 nM T94621 CPJZ24 11584546 IC50 = 696 nM T94621 C0SCK2 11585287 IC50 = 8923 nM T94621 CAP6N0 11588244 IC50 = 8 nM T94621 CMIL86 11590363 Ki > 8400 nM T94621 C6C0VR 11592032 IC50 = 1131 nM T94621 C61KCW 11596252 IC50 = 680 nM T94621 CK61VI 11606572 IC50 = 3706 nM T94621 C20IRX 11606613 IC50 = 1304 nM T94621 C7PA8T 11607451 IC50 = 27 nM T94621 CNA3X5 11608401 IC50 = 6900 nM T94621 C3FQP1 11614515 IC50 = 4 nM T94621 CBEG76 11621110 IC50 = 635 nM T94621 C7P8CI 11622815 IC50 = 9500 nM T94621 CP2R3O 11636277 IC50 = 45 nM T94621 C4YWT2 11636404 IC50 = 6 nM T94621 C9T6SC 11640926 Ki > 8400 nM T94621 C2OC8S 11642946 IC50 = 43 nM T94621 CDY01B 11643074 IC50 = 252 nM T94621 C9RLC8 11643116 IC50 = 77 nM T94621 CP0I2U 11643417 IC50 = 25 nM T94621 CPA5Y7 11650332 IC50 = 184 nM T94621 COR9B8 11650399 IC50 = 16 nM T94621 CBW0A4 11660816 IC50 = 250 nM T94621 C87JQN 11663666 IC50 = 281 nM T94621 C7XEV0 11664023 IC50 = 94.4 nM T94621 CESQ80 11670972 IC50 = 239 nM T94621 C43LDG 11671553 IC50 = 73 nM T94621 CTI6U1 11671757 IC50 = 47 nM T94621 CX1GS0 11672017 IC50 = 16 nM T94621 CON70D 11672049 IC50 = 68 nM T94621 C0V7SU 11675388 IC50 = 2.2 nM T94621 CC5B1E 11681688 IC50 = 16 nM T94621 C0Q7ZW 11688053 IC50 = 400 nM T94621 CU0E8O 11690457 Ki > 10000 nM T94621 C81CLV 11693440 IC50 = 138 nM T94621 C95XBF 11695362 IC50 = 430 nM T94621 CPK2W8 11696113 IC50 = 5 nM T94621 C0NRG1 11703456 IC50 = 8 nM T94621 CB0AP2 11705863 Ki > 10000 nM T94621 CG3RQ4 11708454 IC50 = 290 nM T94621 C3B2HN 11708521 IC50 = 3200 nM T94621 CCK3Q5 11712132 IC50 = 1242 nM T94621 CY8U0T 11713130 IC50 = 90 nM T94621 CM49IK 11715597 IC50 = 920 nM T94621 C0TN5D 11738219 IC50 = 200 nM T94621 CJKC74 11750389 IC50 = 17 nM T94621 C9A6KM 11857236 Ki = 2 nM T94621 CA9ST2 11959186 IC50 = 63 nM T94621 CC7M0D 11959190 IC50 = 50 nM T94621 C39VTW 11959283 IC50 = 63 nM T94621 CQ8U1P 11959284 IC50 = 16 nM T94621 C36HDX 11959286 IC50 = 40 nM T94621 CTE96C 11959310 IC50 = 25 nM T94621 CO0A4K 11959314 Ki = 5 nM T94621 C12CRJ 11959377 IC50 = 200 nM T94621 CUWL12 11959378 IC50 = 25 nM T94621 CVPT94 11959513 IC50 = 316 nM T94621 C5LZ9C 11959550 IC50 = 200 nM T94621 C3UVQ2 11959600 IC50 = 79 nM T94621 C1WDQ0 11959682 IC50 = 20 nM T94621 CMW89V 11959683 IC50 = 20 nM T94621 CA6K4Y 11959684 IC50 = 20 nM T94621 C7RNV1 15602982 IC50 = 280 nM T94621 C3P1ED 15602983 IC50 = 34000 nM T94621 C7N6CQ 15604547 IC50 = 21 nM T94621 CSA02I 15979148 IC50 = 14.6 nM T94621 CBE54Y 15979149 IC50 = 6.7 nM T94621 C9YE7I 15979150 IC50 = 2.8 nM T94621 C92FEN 15979151 IC50 = 10.4 nM T94621 C9QO8U 15979276 IC50 = 10 nM T94621 CFPW41 16007116 Ki > 8400 nM T94621 CZK8V6 16043304 IC50 = 23 nM T94621 C9TU1O 16046126 IC50 > 1000 nM T94621 CKV4G1 16079040 IC50 = 20 nM T94621 CBM80K 16091080 IC50 = 47.7 nM T94621 C7Z4LV 16095343 IC50 = 1950 nM T94621 CHR8G4 16122633 IC50 = 20 nM T94621 C51PSY 16122634 IC50 = 5200 nM T94621 C2RNZ0 16657945 IC50 = 9 nM T94621 C94ONJ 16658020 IC50 = 12000 nM T94621 CSR4V7 16658021 IC50 = 3000 nM T94621 C0O6SY 17751068 IC50 = 8.5 nM T94621 CSK49V 17751069 IC50 = 7 nM T94621 C9C5TV 17751819 IC50 = 6 nM T94621 CWK2H5 21103101 IC50 = 274 nM T94621 CA46OM 21103107 IC50 > 50000 nM T94621 CJXU82 21103111 IC50 = 1877 nM T94621 CF9YE6 21103119 IC50 = 332 nM T94621 C5AR9M 21103197 IC50 = 281 nM T94621 CN1O7X 23647016 IC50 > 50000 nM T94621 CJ3EO0 23647017 IC50 = 1755 nM T94621 CH14KD 23647018 IC50 = 45270 nM T94621 CQ5Z0J 23647019 IC50 = 5407 nM T94621 CT7XW8 23647020 IC50 > 50000 nM T94621 C2JTA3 23647573 IC50 = 5 nM T94621 C83PYS 23647592 IC50 = 9 nM T94621 CI90XG 23647594 IC50 = 21 nM T94621 CWE47K 23647595 IC50 = 45 nM T94621 CICB91 23647596 IC50 = 4 nM T94621 C7W0PE 23647597 IC50 = 4 nM T94621 CTI1F7 23647598 IC50 = 6 nM T94621 CSOG98 23647599 IC50 = 19 nM T94621 CJAI42 23647600 IC50 = 51 nM T94621 CUX75S 23647601 IC50 = 37 nM T94621 CUX5O6 23647602 IC50 = 5 nM T94621 CA4LE6 23647603 IC50 = 8 nM T94621 CGS7Q3 23647604 IC50 = 3 nM T94621 CH89JW 23647605 IC50 = 5 nM T94621 CLDV63 23647606 IC50 = 5 nM T94621 C2BHO1 23658108 IC50 = 25 nM T94621 CL8M1D 23658126 IC50 = 5 nM T94621 CC97WO 23658173 IC50 = 70 nM T94621 CSJ34W 24701731 IC50 = 270 nM T94621 C7YG1N 24759534 IC50 = 23000 nM T94621 C7R9TA 24762195 IC50 = 8 nM T94621 CQNP54 24764449 IC50 = 25000 nM T94621 CW3JR8 24783593 IC50 = 14 nM T94621 C05MQY 24783594 IC50 = 35 nM T94621 C93TIM 24786152 IC50 = 12 nM T94621 CSY9Z6 24788164 IC50 = 11 nM T94621 CFR62V 24788432 IC50 = 12 nM T94621 C2JNI3 24788623 IC50 = 17 nM T94621 CMR7F1 24788739 IC50 = 15 nM T94621 CY1ZS7 24803305 Ki = 3 nM T94621 C2ANO6 24804134 Ki = 8 nM T94621 CSH8A5 24804780 Ki = 6 nM T94621 CUTH13 24805273 IC50 = 125 nM T94621 C0AO5R 24828715 IC50 = 110000 nM T94621 C1H2AM 24828716 IC50 = 246 nM T94621 CU9E4W 24828717 IC50 = 12 nM T94621 C5U2ZM 24828854 IC50 = 3 nM T94621 CQ4G2E 24828855 IC50 = 7 nM T94621 C57SYK 24829098 IC50 = 25 nM T94621 C3YLM1 24829099 IC50 = 71 nM T94621 CM5AX9 24829102 IC50 = 25 nM T94621 CY97JK 24829220 IC50 = 7 nM T94621 CT7QD8 24829222 IC50 = 25 nM T94621 C5WS6R 24894100 IC50 = 48 nM T94621 CV5IE4 24963049 Ki = 1 nM T94621 C9YN2Q 24967131 IC50 > 10000 nM T94621 CLJ2N0 24971386 IC50 = 1299 nM T94621 CC7B8W 24971387 IC50 = 1709 nM T94621 CCWV70 24971388 IC50 = 1381 nM T94621 CSE34D 24971389 IC50 = 1160 nM T94621 C5NFP2 24971390 IC50 = 1514 nM T94621 C0B9HE 24971391 IC50 = 17470 nM T94621 CX1U6V 24971392 IC50 = 1792 nM T94621 C3JT8Q 24971393 IC50 = 494 nM T94621 C0PFZ7 24992842 IC50 = 35 nM T94621 CC61ER 24993160 IC50 = 46 nM T94621 CT81XK 24993161 IC50 = 44 nM T94621 CZK9Q1 24993162 IC50 = 5.5 nM T94621 CK0NZ8 24993163 IC50 = 27 nM T94621 CQ9BF6 24993164 IC50 = 15 nM T94621 C71EOU 24993165 IC50 = 90 nM T94621 C1Y3TF 24993166 IC50 = 20 nM T94621 CA9F3Y 25023714 IC50 = 1000 nM T94621 C8Z4PI 25023715 IC50 = 3980 nM T94621 CV96QX 25023716 IC50 = 2340 nM T94621 C5INV4 25023717 IC50 = 2510 nM T94621 CPOH02 25023718 IC50 = 10000 nM T94621 C6F7RD 25023719 IC50 = 2570 nM T94621 C1JEU6 25023729 IC50 = 9 nM T94621 C14NAT 25023731 IC50 = 20 nM T94621 C81XKW 25023732 IC50 = 4 nM T94621 CFH80B 25023733 IC50 = 13 nM T94621 CR8JP7 25023735 IC50 = 13 nM T94621 C4W7LY 25023736 IC50 = 6 nM T94621 CA6QU5 25023737 IC50 = 5 nM T94621 COV3Q4 25061501 IC50 = 9 nM T94621 C8NR9H 25170562 IC50 = 6 nM T94621 CS9LC3 25170563 IC50 = 22 nM T94621 CN8YZ4 25170991 IC50 = 29 nM T94621 CHN5O0 25190977 IC50 = 19 nM T94621 COWB90 25221040 IC50 = 130 nM T94621 CC25TV 25222706 IC50 = 13 nM T94621 C1IG7E 25243798 IC50 > 10000 nM T94621 CH65JV 25243799 IC50 > 10000 nM T94621 CBQO98 42602095 IC50 = 40 nM T94621 CJ61SE 42602096 IC50 = 23 nM T94621 CI42XG 42602097 IC50 = 30 nM T94621 CD2AH4 42602175 IC50 = 24 nM T94621 CSWA85 42602176 IC50 = 46 nM T94621 C1LUN4 42602178 IC50 = 14 nM T94621 C8O3EA 42602260 IC50 = 22 nM T94621 C93NKL 42602264 IC50 = 15 nM T94621 C59CDG 44389260 IC50 = 157 nM T94621 CEP4T0 44422924 IC50 = 10 nM T94621 C0PEK6 44426856 IC50 = 31 nM T94621 COP8A3 44449880 IC50 = 42 nM T94621 CMC82Z 44449900 IC50 = 1476 nM T94621 C3APO5 44449908 IC50 = 210 nM T94621 CA85HS 44449909 IC50 = 981 nM T94621 C4QJK8 44449942 IC50 = 1600 nM T94621 C0ICB5 44449973 IC50 = 280 nM T94621 CE15WY 44449975 IC50 = 900 nM T94621 CEWB75 44450002 IC50 = 260 nM T94621 CDEJ84 44450004 IC50 = 1075 nM T94621 C8OG1V 44517709 IC50 = 1500 nM T94621 C1EVH2 44560678 IC50 = 827 nM T94621 CI58CZ 44560679 IC50 = 224 nM T94621 CC4Z5M 44560681 IC50 = 165 nM T94621 CWOM65 44560715 IC50 = 40 nM T94621 C7YCO3 44560716 IC50 = 80 nM T94621 C5X7PO 44560717 IC50 = 130 nM T94621 COTH35 44560718 IC50 = 84 nM T94621 C6J0ZC 44560719 IC50 = 180 nM T94621 CL0A2D 44560720 IC50 = 140 nM T94621 CR8K0X 44560724 IC50 = 185 nM T94621 CE08JD 44560725 IC50 = 146 nM T94621 CSX84T 44560726 IC50 = 92 nM T94621 C1O0IG 44560727 IC50 = 43 nM T94621 CB7X4S 44560728 IC50 = 192 nM T94621 C94LIO 44560729 IC50 = 190 nM T94621 C3UQ8C 44560730 IC50 = 116 nM T94621 C8OD4F 44560731 IC50 = 225 nM T94621 CLB20U 44560732 IC50 = 230 nM T94621 CGY1X7 44561054 IC50 = 29 nM T94621 CZK43G 44561055 IC50 = 223 nM T94621 C4WLX8 44561056 IC50 = 421 nM T94621 CXC8I3 44561057 IC50 = 23 nM T94621 CS0QZ4 44561058 IC50 = 539 nM T94621 C1QG9P 44561059 IC50 = 3570 nM T94621 C9MTS4 44561060 IC50 = 59 nM T94621 CZ9L8F 44572052 IC50 = 24.1 nM T94621 CIV48S 44572053 IC50 = 483.3 nM T94621 CFVA91 44572054 IC50 = 55.1 nM T94621 CZE8M9 44572055 IC50 = 77.9 nM T94621 C0DJS1 44591843 Ki = 4 nM T94621 CX52YW 44591844 Ki = 4 nM T94621 C1LS6V 44591845 Ki = 16 nM T94621 CSZ5R9 44592438 IC50 = 500 nM T94621 C6X7FC 44592501 Ki = 40 nM T94621 CTS95L 44592502 Ki = 40 nM T94621 CSKZ16 44592503 IC50 = 8 nM T94621 COY57J 44592504 Ki = 0.63 nM T94621 C3CDV8 44592505 Ki = 2 nM T94621 CJK7L8 45141615 IC50 = 19 nM T94621 CUEX28 45141616 IC50 = 84 nM T94621 C7XZI3 45141617 IC50 > 1000 nM T94621 CZC94D 45141618 IC50 = 35 nM T94621 CY8DC7 45141619 IC50 = 16 nM T94621 C5N4FO 45141620 IC50 = 18 nM T94621 CSB9Q2 45141621 IC50 = 69 nM T94621 C9BXC0 45141812 IC50 = 7 nM T94621 CEU36T 45141813 IC50 = 36 nM T94621 CLED29 45141814 IC50 = 14 nM T94621 CC16ZH 45141815 IC50 = 11 nM T94621 CM57PW 45141816 IC50 = 29 nM T94621 CC3R8E 45141817 IC50 = 210 nM T94621 CQ7OZ9 45142021 IC50 = 4.9 nM T94621 C01CFQ 45142022 IC50 = 5.7 nM T94621 C7FS2V 45142023 IC50 = 11 nM T94621 CYBD69 45142024 IC50 = 8 nM T94621 CR37UP 45142025 IC50 = 4 nM T94621 CU2K8B 45142026 IC50 = 25 nM T94621 CE4D3F 45142255 IC50 = 31 nM T94621 CLCU70 45142256 IC50 = 12 nM T94621 CJQ28R 45142257 IC50 = 52 nM T94621 CJIA74 45142258 IC50 = 12 nM T94621 C1V2YL 45142259 IC50 = 58 nM T94621 CQ5SD4 46190876 IC50 = 39 nM T94621 CY3HW5 46224684 IC50 = 4200 nM T94621 CB5H9C 46225574 IC50 = 31 nM T94621 C8M1DT 46225589 IC50 = 6 nM T94621 C60XUQ 46226079 IC50 = 15 nM T94621 C5PCH8 46226080 IC50 = 15 nM T94621 C6UD1Y 46226095 IC50 = 250 nM T94621 C7IF4T 46226096 IC50 = 63 nM T94621 CUDZ46 46226135 IC50 = 6300 nM T94621 C0P4CT 46226136 IC50 = 12 nM T94621 CPH49S 46226137 IC50 = 7 nM T94621 CM5X8B 46226156 IC50 = 15 nM T94621 C64TVL 46226417 IC50 = 25 nM T94621 CLS29B 46872626 IC50 > 10000 nM T94621 C2O8RZ 46886323 IC50 > 1000 nM T94621 CM8RX4 46886549 Ki = 17 nM T94621 C70BLN 46886550 IC50 = 50 nM T94621 CCV96R 46886665 Ki = 39 nM T94621 CJ2E9Q 46929857 IC50 > 25000 nM T94621 CC1Y0M 52941299 IC50 = 4951 nM T94621 CDT94U 52941495 IC50 = 1485 nM T94621 C9UF6K 52941555 IC50 = 433 nM T94621 CYM80Q 52942489 IC50 = 37826 nM T94621 CS09YT 52942516 IC50 = 5027 nM T94621 CQ08WT 52942668 IC50 = 1288 nM T94621 CHW04J 52943916 IC50 = 630 nM T94621 CY8BV4 52944892 IC50 = 707 nM T94621 CEM95A 52946401 IC50 = 5586 nM T94621 CKE3C7 52946402 IC50 = 1067 nM T94621 C3Q4CU 52947490 IC50 = 8362 nM T94621 CR9E1Z 52947590 IC50 = 26500 nM T94621 CE81HA 52950003 IC50 = 279 nM T94621 C3TU8R 52950063 IC50 = 872 nM T94621 C7MC5G 52950205 IC50 = 4371 nM T94621 C8NA4L 53384644 IC50 > 30000 nM T94621 CO6B0E 54583043 IC50 > 10000 nM T94621 C3PGE2 54585958 IC50 > 10000 nM T94621 CV7HJ8 54585959 IC50 > 10000 nM T94621 CPC5D2 56603995 IC50 = 8 nM T94621 CFP56A 56604013 IC50 = 8 nM T94621 CM8JX1 56604907 IC50 = 25000 nM T94621 CN9QD7 56643097 IC50 > 10000 nM T94621 CT4E8R 56832546 IC50 = 3300 nM T94621 CS7U9L 56965952 IC50 = 18 nM T94621 CQ57PE 57345536 IC50 = 3021 nM T94621 CQP7E0 57750290 IC50 = 31 nM T94621 CNBO65 57750312 IC50 = 36 nM T94621 C2F9DS 57750315 IC50 = 159 nM T94621 CZ08KN 57750321 IC50 = 96 nM T94621 CUY8T6 57750329 IC50 = 709 nM T94621 CK4W1L 57750342 IC50 = 30 nM T94621 CM5X9L 57750343 IC50 = 836 nM T94621 CBY5E4 57750369 IC50 = 42 nM T94621 CSI9Y4 57750382 IC50 = 210 nM T94621 C6GH7X 57750391 IC50 = 190 nM T94621 CL7CW0 57750402 IC50 = 130 nM T94621 CA4G5W 57750407 IC50 = 13 nM T94621 CM7XL6 57750408 IC50 = 20 nM T94621 CY4Z8R 57750418 IC50 = 344 nM T94621 C87LKR 58191080 IC50 = 4 nM T94621 CZPF92 58191081 IC50 = 6 nM T94621 CZA32V 58344912 IC50 = 700 nM T94621 CPVF85 58344916 IC50 = 660 nM T94621 CD3LX9 58344922 IC50 = 15 nM T94621 CS8ZY7 58344924 IC50 = 25 nM T94621 C89NVR 58344941 IC50 = 47 nM T94621 CYK74H 58344983 IC50 = 32 nM T94621 CRJ47B 58345005 IC50 = 16000 nM T94621 CIOV02 58345019 IC50 = 800 nM T94621 CY62SG 58345029 IC50 = 30 nM T94621 CM5HE1 58345070 IC50 = 130 nM T94621 CO18NP 58345151 IC50 = 35 nM T94621 CV61YJ 58345169 IC50 = 51000 nM T94621 CW6SC9 58345215 IC50 = 20000 nM T94621 CFLZ87 58345232 IC50 = 24 nM T94621 CYBT41 58345302 IC50 = 80 nM T94621 C4PE7X 58345314 IC50 = 27 nM T94621 C8X3WB 58458198 IC50 = 4177 nM T94621 C20XPF 58458267 IC50 > 2000 nM T94621 CP85TJ 58458278 IC50 = 6 nM T94621 CT79LH 58458379 IC50 = 356 nM T94621 CXJ63M 59603829 IC50 > 100000 nM T94621 CQEU96 59603842 IC50 = 430 nM T94621 CPVD45 59670809 IC50 = 33 nM T94621 C32WHR 59670989 IC50 = 24 nM T94621 CDWQ04 59671004 IC50 = 31 nM T94621 C43HZT 59671085 IC50 = 249 nM T94621 C0BRA5 59671144 IC50 = 66 nM T94621 CEYW16 59671148 IC50 = 10 nM T94621 C50NWX 59671151 IC50 = 3 nM T94621 CZH4W5 59671179 IC50 = 18 nM T94621 C8FY0G 59671180 IC50 = 17 nM T94621 COH62U 60097413 IC50 > 5000 nM T94621 C1MR8Q 60097495 IC50 > 10000 nM T94621 CC3MB4 60155179 IC50 = 9300 nM T94621 C9QB8G 60155270 IC50 = 1900 nM T94621 CM6NF2 60155627 IC50 = 3500 nM T94621 C62SQG 60155628 IC50 = 24 nM T94621 COS39T 60155629 IC50 = 33 nM T94621 CG6XQ3 67161715 IC50 = 477 nM T94621 CNXU89 67162253 IC50 = 311 nM T94621 CV63UL 67240318 IC50 > 10000 nM T94621 CP8OI2 67304551 IC50 = 5300 nM T94621 CY76UR 67305743 IC50 = 4.5 nM T94621 C3UKG8 67312397 IC50 = 3.2 nM T94621 CM6TZ3 67312506 IC50 = 2.5 nM T94621 C5DGR9 69036886 IC50 = 10000 nM T94621 CS8UF1 70675988 IC50 = 6 nM T94621 C2W5BX 70675991 IC50 = 2005 nM T94621 CUJA60 70676312 IC50 = 6 nM T94621 CRBW21 70676316 IC50 = 30 nM T94621 CGX49K 70676464 IC50 = 5 nM T94621 C1IEJ2 70789254 IC50 = 66000 nM T94621 C8T7ZP 70789255 IC50 = 9500 nM T94621 CKT60L 71455860 Ki > 8000 nM T94621 C9DIK2 71512060 IC50 > 10000 nM T94621 CQV96E 71583048 IC50 = 8111 nM T94621 CSPR52 71583049 IC50 = 16498 nM T94621 CNT5F3 71583050 IC50 = 805 nM T94621 CH7I0W 71583051 IC50 = 8578 nM T94621 CXSI14 71718330 IC50 > 100000 nM T94621 C1TM3P 71720141 IC50 > 100000 nM T94621 CJ2T9E 76332983 IC50 > 10000 nM T94621 C1HW4B 89735655 IC50 = 2500 nM T94621 CQCX41 118737057 IC50 > 10000 nM T94621 C9J4ES 135503073 IC50 = 8 nM T94621 CK94UW 136036657 IC50 = 83 nM T94621 CO16JK 136099766 IC50 = 188 nM T94621 C3ZS9L 136099767 IC50 = 284 nM T94621 CLB4O7 136099768 IC50 = 98 nM T94621 CC73PA 138911338 IC50 = 1.2 nM T94621 CSU93V 155077019 IC50 = 0.54 nM T94621 C2MD1Q 155513187 IC50 > 10000 nM T94621 C86HPW 155518524 IC50 = 21000 nM T94621 CL5DR0 155525783 IC50 < 0.64 nM T94621 CHS21A 155553831 IC50 = 14 nM T94621 CG95WV 155563831 IC50 = 2.8 nM T94621 CEIW13 155566807 IC50 = 79 nM T94621 D00ERW 44444843 Ki = 4800 nM T94621 D00HVA 11624601 Ki > 8400 nM T94621 D05APZ 135398501 IC50 = 210 nM T94621 D09FFE 449241 IC50 = 590 nM T94621 D0I1FJ 11393719 IC50 = 741 nM T94621 D0L2WP 46225540 IC50 = 12 nM T94621 D0OX1T 10172943 IC50 = 30 nM T94621 D0Q3NG 11715520 Ki > 8400 nM T94621 D0R2WK 16038120 Ki > 10000 nM T94621 D0S7IE 11658882 Ki > 8400 nM T94621 D0V6GX 11311693 IC50 = 20 nM T59720 C9G0HL 10533268 Ki = 35 nM T59720 C0QN5G 10606215 Ki = 35 nM T59720 C4IZ1Y 10820377 Ki = 35 nM T59720 CA50FN 56662663 Ki = 35 nM T59720 CH3SW7 56679684 Ki = 35 nM T43031 D0E3TC 44259 IC50 = 18.4 nM T43031 C1SVD2 2132479 IC50 = 3500 nM T43031 C18HKQ 9885748 IC50 = 77000 nM T43031 CACS26 11561968 Ki > 2000 nM T43031 CU0E8O 11690457 Ki > 2000 nM T43031 CKV4G1 16079040 IC50 = 500 nM T43031 CL81VC 21100709 IC50 = 11500 nM T43031 CZ3XP5 46926535 IC50 = 2600 nM T43031 C75GBE 49837568 IC50 = 22500 nM T43031 CEQN27 52936621 Ki > 1000 nM T43031 CT4E8R 56832546 IC50 = 14000 nM T43031 C1MR8Q 60097495 IC50 > 1000 nM T43031 CV63UL 67240318 IC50 = 630 nM T43031 CXSI14 71718330 IC50 = 83000 nM T43031 C1TM3P 71720141 IC50 = 83000 nM T43031 CJ2T9E 76332983 IC50 > 10000 nM T43031 C07EKN 138454794 IC50 > 10000 nM T43031 C0BU2E 145954767 IC50 > 10000 nM T43031 C2MD1Q 155513187 IC50 > 10000 nM T43031 D0K0UJ 49837564 IC50 = 170 nM T55922 D05FFR 5351154 Ki > 1000 nM T55922 CD0Y2A 118705586 Ki = 1070000 nM T55922 CD64YM 118725236 Ki = 1207000 nM T55922 C4ZJU9 239269 IC50 > 180000 nM T55922 CL14FJ 240808 IC50 > 180000 nM T55922 C9BOU0 240809 IC50 > 180000 nM T55922 CD3MU4 388060 IC50 > 180000 nM T55922 CG8Y0J 463012 IC50 > 180000 nM T55922 C1EPW6 476291 IC50 = 1500 nM T55922 CWN21X 608203 IC50 > 180000 nM T55922 CHU71V 2766291 IC50 > 180000 nM T55922 C3KV6A 11742879 Ki = 21200 nM T55922 C7HG1T 15218331 Ki = 20600 nM T55922 C1M3XT 19754189 IC50 > 180000 nM T55922 C05HNS 25181313 IC50 = 400 nM T55922 CQ39IJ 25183746 IC50 = 31000 nM T55922 CV90QL 25231313 IC50 = 3000 nM T55922 CTN16A 25231650 IC50 = 4000 nM T55922 C7NB0S 25231818 IC50 = 170 nM T55922 CIF3B2 25231819 IC50 = 440000 nM T55922 CH84SG 25231821 IC50 = 500000 nM T55922 CDS82O 25232183 IC50 = 49 nM T55922 CP1DT0 25233591 IC50 = 88000 nM T55922 C5BL4R 25233958 IC50 = 157000 nM T55922 C2EMK0 29066960 IC50 > 180000 nM T55922 CHB02E 44564175 IC50 = 7 nM T55922 C1L3WI 44564176 IC50 = 86 nM T55922 CE0JM4 44564196 IC50 = 11 nM T55922 CMWC14 44564197 IC50 = 5 nM T55922 CAID84 44564238 IC50 = 15 nM T55922 CFB5I1 44564239 IC50 = 18 nM T55922 CB7U4V 44564271 IC50 = 7000 nM T55922 CS43LM 44564338 IC50 = 70000 nM T55922 C57HRM 44564339 IC50 = 420000 nM T55922 C9Q3ZV 45097405 IC50 > 180000 nM T55922 C8UP6J 56919646 IC50 > 180000 nM T55922 CNI72Y 56919796 IC50 > 180000 nM T55922 C6A4KE 56919816 IC50 > 180000 nM T55922 C8I4ZA 56919856 IC50 > 180000 nM T55922 COU16Q 56920121 IC50 > 180000 nM T55922 CKLS86 56920454 IC50 > 180000 nM T55922 C8B4NQ 56920865 IC50 > 180000 nM T55922 C4T8JN 56921130 IC50 > 180000 nM T55922 C5CHU3 56921153 IC50 > 180000 nM T55922 CZHJ85 56921749 IC50 > 180000 nM T55922 C4U2XL 56921808 IC50 > 180000 nM T55922 COC17L 56922155 IC50 > 180000 nM T55922 C84CMO 56922551 IC50 > 180000 nM T55922 CUB52I 56923076 IC50 > 180000 nM T55922 CFG3V8 61710896 IC50 > 180000 nM T55922 C0Q8VJ 71460033 Ki = 3800 nM T55922 CA5VM1 80647643 IC50 > 180000 nM T55922 CHF61P 80761654 IC50 > 180000 nM T55922 C5JT8K 80768222 IC50 > 180000 nM T55922 C1B3TQ 80768523 IC50 > 63000 nM T55922 CFB2V6 80768610 IC50 > 180000 nM T55922 CGM4L1 100765007 IC50 > 180000 nM T55922 C8AF7O 104032679 IC50 > 180000 nM T55922 CV6FI3 107371081 IC50 > 180000 nM T55922 CW9RE8 113977178 IC50 > 160000 nM T55922 CIZ98T 114563625 IC50 > 180000 nM T55922 CP68ZQ 118725161 Ki = 21200 nM T55922 CUX9J4 118725180 Ki = 19600 nM T55922 CI9ZG7 118725204 Ki = 7200 nM T55922 CTB96Z 118725211 IC50 = 9000 nM T55922 CG8LY5 118725234 Ki = 18000 nM T55922 CI7C4Q 118725235 Ki = 669000 nM T55922 CZ4AP8 118725238 Ki = 478000 nM T55922 CQI0V5 118725241 Ki = 415000 nM T55922 CX13CP 118725243 Ki = 960000 nM T55922 CL3QZ8 118725244 IC50 = 178600 nM T55922 CAQH86 118725250 IC50 = 204800 nM T55922 CMS1X0 137632229 IC50 > 180000 nM T55922 CA6JL1 137632834 IC50 > 180000 nM T55922 CS1V5F 137632899 IC50 > 180000 nM T55922 CVC92M 137634051 IC50 > 180000 nM T55922 C82GYX 137634161 IC50 > 180000 nM T55922 CX84ME 137634646 IC50 > 180000 nM T55922 CT85ZK 137635286 IC50 > 180000 nM T55922 CGWV42 137635709 IC50 > 180000 nM T55922 C0D3HO 137635782 IC50 > 180000 nM T55922 C9ANK4 137635823 IC50 > 180000 nM T55922 CIKN81 137637985 IC50 > 63000 nM T55922 C8LO3S 137638905 IC50 > 180000 nM T55922 C7IWK8 137639930 IC50 > 180000 nM T55922 C6K3NC 137640514 IC50 > 180000 nM T55922 CD9HO6 137641254 IC50 > 21000 nM T55922 CK4NM7 137642459 IC50 > 180000 nM T55922 CT9Z2B 137642510 IC50 > 180000 nM T55922 CP05EG 137642600 IC50 > 63000 nM T55922 CPL3I7 137642845 IC50 = 44000 nM T55922 CF3W1S 137644197 IC50 > 63000 nM T55922 CO2ZG3 137645098 IC50 > 180000 nM T55922 CZ39RI 137645795 IC50 > 180000 nM T55922 CR2G4T 137646814 IC50 > 63000 nM T55922 C5D8MS 137647022 IC50 > 180000 nM T55922 CYA0M8 137648601 IC50 > 180000 nM T55922 C8J6EA 137648725 IC50 > 180000 nM T55922 C5HQ3N 137648979 IC50 > 21000 nM T55922 C4XUM8 137649315 IC50 > 21000 nM T55922 CNK2S4 137650167 IC50 > 180000 nM T55922 CE8ID4 137650445 IC50 > 180000 nM T55922 C9K4XH 137651053 IC50 > 21000 nM T55922 C75RCW 137651145 IC50 > 7000 nM T55922 C4C9DG 137651239 IC50 > 180000 nM T55922 CD23LP 137651376 IC50 > 63000 nM T55922 C03QHT 137651433 IC50 > 180000 nM T55922 C0TO6G 137651822 IC50 > 180000 nM T55922 CQE98H 137652324 IC50 > 180000 nM T55922 CHM69W 137652349 IC50 > 180000 nM T55922 CE57MT 137652443 IC50 > 180000 nM T55922 C46JEQ 137652753 IC50 > 180000 nM T55922 CFCI38 137652950 IC50 > 180000 nM T55922 C4GMS8 137653057 IC50 > 180000 nM T55922 CPZ58N 137653090 IC50 > 21000 nM T55922 CGK5Y1 137653360 IC50 > 180000 nM T55922 CSQF12 137653636 IC50 > 180000 nM T55922 CP8TJ0 137654766 IC50 > 21000 nM T55922 C75NWC 137655212 IC50 > 180000 nM T55922 CR6N5Y 137656925 IC50 > 21000 nM T55922 C9PJD2 137657088 IC50 > 180000 nM T55922 C5Q0YO 137657983 IC50 > 180000 nM T55922 CJ4M7L 137658244 IC50 > 180000 nM T55922 C3RO8E 137659106 IC50 > 180000 nM T55922 C6BN1M 137659420 IC50 > 63000 nM T55922 CBXA79 137659429 IC50 > 63000 nM T55922 CYD2N8 137659438 IC50 > 180000 nM T55922 C71FOJ 137660126 IC50 > 180000 nM T55922 C89UTS 137660314 IC50 > 63000 nM T55922 CPZ9E8 137660942 IC50 > 180000 nM T55922 CD1Y9L 137660985 IC50 > 180000 nM T55922 C4QM7T 137662328 IC50 > 180000 nM T55922 D03OLX 25231309 IC50 = 9000 nM T55922 D0I7IA 25231315 IC50 = 5000 nM T55922 D0P5YR 446204 IC50 = 55 nM T55922 D0YM6B 25231308 IC50 = 600 nM T58130 CN8XM2 5311263 EC50 = 8.1 nM T58130 CLS96Y 6419701 EC50 = 83.18 nM T58130 COZF72 10322404 EC50 = 2.692 nM T58130 C7QRT8 11648176 EC50 = 3.8 nM T58130 CV86RF 44368508 EC50 = 4.898 nM T58130 C85ANH 46213949 IC50 > 8000 nM T58130 CET63X 46223906 EC50 = 3.3 nM T58130 C57TYK 71569053 EC50 = 3.8 nM T58130 CSN3I7 71569056 EC50 = 2.4 nM T58130 CPT5S2 71718248 EC50 = 4.467 nM T58130 CKC4U7 71719457 EC50 = 4.898 nM T58130 C5P1CQ 71720690 EC50 = 3.467 nM T58130 CG65XZ 122191108 Ki = 170 nM T58130 CWQ8Y3 122191544 IC50 = 266 nM T58130 D05TVG 23682233 Ki = 170 nM T58130 D0X0UR 5497152 EC50 = 570 nM T17345 D01KKQ 135400182 IC50 = 21000 nM T17345 D0AO5H 5578 Ki = 0.006 nM T17345 D0C0SK 4993 Ki = 8 nM T17345 D0H0KB 5070 IC50 = 312000 nM T17345 D0M4VM 5320 IC50 = 18000 nM T17345 D0SV8E 126941 Ki = 0.00034 nM T17345 D0Y4GO 135410875 Ki = 7 nM T17345 D0Y7TS 5583 IC50 < 1 nM T17345 D04LBC 213043 IC50 = 8 nM T17345 D09AYQ 54369 Ki = 0.025 nM T17345 D05HCO 177894 Ki = 0.0003 nM T17345 D05AHQ 68916 Ki = 58.88 nM T17345 D06YIB 135436405 IC50 > 100000 nM T17345 D0D2RN 169371 Ki = 0.0018 nM T17345 D0FC5T 21453 IC50 = 530 nM T17345 D0N3XT 57030 IC50 = 1.8 nM T17345 CND0P2 1881 Ki = 4.5 nM T17345 C7OTP8 3439 IC50 = 220 nM T17345 CU2C4N 3534 IC50 = 70000 nM T17345 C8Y3OG 3537 IC50 = 2000 nM T17345 CEJF30 19931 Ki = 1659.59 nM T17345 C1F2TO 25889 Ki = 110 nM T17345 CY85FK 38778 Ki = 77.62 nM T17345 CRV0E5 72468 IC50 = 1000 nM T17345 CZ8JM5 72509 IC50 = 2.7 nM T17345 C87TYO 72934 IC50 = 15 nM T17345 C7SXL6 87152 IC50 = 1040000 nM T17345 CJ19OK 101067 Ki = 9.6 nM T17345 C8OGL7 102185 IC50 = 9400 nM T17345 C1Q8JR 121750 Ki = 7.7 nM T17345 C4HSB8 125843 IC50 = 1.35 nM T17345 CZA4M3 158351 IC50 = 220 nM T17345 CRQ24H 160203 Ki = 22.39 nM T17345 CZM82G 269322 IC50 = 3.9 nM T17345 C82AVZ 275733 IC50 = 3.8 nM T17345 C5JO7S 316019 IC50 = 3000 nM T17345 C3BRV9 317332 IC50 = 2700 nM T17345 CV20SE 324351 IC50 = 4.1 nM T17345 CPI45H 324352 IC50 = 8.6 nM T17345 CWV02U 324357 IC50 = 5.8 nM T17345 CY8C9L 329597 IC50 = 25000 nM T17345 C9GDJ6 353015 Ki = 0.00089 nM T17345 C3QH5B 354441 Ki = 218.78 nM T17345 CE7IH3 354768 IC50 = 19 nM T17345 CHA7L8 360682 Ki = 0.00035 nM T17345 CT64FM 375312 IC50 = 5.8 nM T17345 CC3ZE0 381233 IC50 = 11.6 nM T17345 C7VFS0 381234 IC50 = 11.4 nM T17345 C3F5KM 382165 IC50 = 8.7 nM T17345 CT51LK 393599 Ki = 0.0004 nM T17345 C8WO4J 403898 Ki = 42000 nM T17345 CTO2D8 404585 Ki = 100 nM T17345 C2IZ4Q 405137 Ki = 1800 nM T17345 C0MKV6 405140 Ki = 600 nM T17345 CDC2L4 406510 Ki = 4000 nM T17345 C25WDV 406511 Ki = 4000 nM T17345 C58ZQB 406512 Ki = 3000 nM T17345 CU4O0N 407233 Ki = 93.33 nM T17345 CD27CT 407235 Ki = 70 nM T17345 C5E7QX 429008 IC50 = 740 nM T17345 C6P2YK 444617 IC50 = 8500 nM T17345 CS9OU4 447021 IC50 = 26 nM T17345 CTXS72 447022 IC50 = 2900 nM T17345 C65ECP 448780 Ki = 5200 nM T17345 CT4N6R 456183 Ki = 6 nM T17345 CYC5M0 456204 IC50 = 4.7 nM T17345 CU1IP4 456205 IC50 < 100 nM T17345 C5VDE1 456216 IC50 = 3900 nM T17345 C1GU8M 456245 IC50 = 820 nM T17345 CD83KY 456272 IC50 = 440 nM T17345 CA6RC1 456306 IC50 = 2700 nM T17345 CQ61JH 456893 IC50 = 5 nM T17345 CEQ98S 456897 IC50 = 18200 nM T17345 CI10YF 457336 IC50 = 150 nM T17345 CHUR38 457342 IC50 = 5.5 nM T17345 CB2ZR6 457343 IC50 = 300 nM T17345 CBD80Z 457349 IC50 = 2300 nM T17345 CX4L1I 457350 IC50 = 1000 nM T17345 C7SZQ6 457353 IC50 = 142 nM T17345 C23EKX 457354 IC50 = 5.1 nM T17345 CBDY12 457370 IC50 = 2600 nM T17345 C81HJP 457371 IC50 = 31000 nM T17345 C53LNC 457372 IC50 = 750 nM T17345 CSWJ43 457373 IC50 = 730 nM T17345 CI17EV 457374 IC50 > 10000 nM T17345 C38SDU 457375 IC50 > 10000 nM T17345 CQY5L9 457376 IC50 > 10000 nM T17345 CMI8V4 457377 IC50 > 10000 nM T17345 CM5JA3 459880 IC50 = 370 nM T17345 CFQ2A9 459881 IC50 = 1000 nM T17345 CW1Q3Y 459887 IC50 = 710 nM T17345 C9YRU0 460024 IC50 = 57 nM T17345 CT9FW6 461920 Ki = 10.2 nM T17345 C03TKX 462111 IC50 = 17 nM T17345 CM4T5X 462117 IC50 = 10 nM T17345 C97EVZ 462118 IC50 = 28000 nM T17345 CHI3D7 462119 IC50 = 28000 nM T17345 C08HAR 462121 IC50 = 26000 nM T17345 C4SOE5 462122 IC50 = 27000 nM T17345 CUO54Z 462123 IC50 = 11 nM T17345 CS04OY 462124 IC50 = 25000 nM T17345 C7DI1F 462125 IC50 = 140 nM T17345 C8WYK9 462127 IC50 = 1400 nM T17345 C6NS9C 462129 IC50 = 50 nM T17345 C4AI1C 462134 IC50 = 3.6 nM T17345 C0EH1R 462466 Ki = 42.66 nM T17345 C8YC0H 462467 Ki = 134.9 nM T17345 CAHX06 462469 Ki = 302 nM T17345 CINY32 462582 IC50 = 2400 nM T17345 C8F9IM 462583 IC50 = 3900 nM T17345 C8QJT5 462584 IC50 = 550 nM T17345 CC65NE 462585 IC50 > 10000 nM T17345 CO46NQ 462587 IC50 = 4300 nM T17345 C62CHU 462589 IC50 = 2100 nM T17345 CTO26P 462590 IC50 = 3100 nM T17345 CQ4DV2 462591 IC50 = 2000 nM T17345 CJ4H0N 462592 IC50 = 2600 nM T17345 C0W2ZP 462593 IC50 = 24000 nM T17345 CBM4S2 462594 IC50 = 33000 nM T17345 C5Z4WX 462595 IC50 = 320 nM T17345 CO05RB 462596 IC50 = 180 nM T17345 C7XI6R 462597 IC50 = 3500 nM T17345 CV80TA 462598 IC50 = 4100 nM T17345 CS1AR6 462599 IC50 = 4400 nM T17345 C74WHR 462600 IC50 = 1300 nM T17345 C3HUT1 462601 IC50 = 400 nM T17345 CEW0T1 462602 IC50 = 270 nM T17345 C52FZM 462603 IC50 = 92 nM T17345 C8PC9F 462604 IC50 = 4300 nM T17345 C7ZJP3 462605 IC50 = 9100 nM T17345 CXW5K6 462606 IC50 = 820 nM T17345 C59MPI 462607 IC50 = 30 nM T17345 CK60HY 463731 IC50 = 990 nM T17345 CO3N7T 463890 IC50 = 12 nM T17345 CVK3W9 463891 IC50 = 7.1 nM T17345 CV4Q2D 463908 IC50 = 1200 nM T17345 C0XBM2 464022 IC50 = 590 nM T17345 C9PX5G 464023 IC50 = 500 nM T17345 C87RIT 464024 IC50 = 850 nM T17345 CMN7V4 464028 IC50 = 6100 nM T17345 CLC49E 464033 IC50 = 440 nM T17345 C6Z1YM 464034 IC50 = 420 nM T17345 C4H1FO 464035 IC50 = 36 nM T17345 CC80XF 464040 IC50 = 10 nM T17345 CRF85I 464992 IC50 = 27 nM T17345 CX8Y6N 464994 IC50 = 670 nM T17345 CCD18G 466230 IC50 = 6.7 nM T17345 CIR4Z5 466231 IC50 = 2500 nM T17345 CZI41B 467890 Ki = 87 nM T17345 CQB5F2 467891 Ki = 29 nM T17345 C0HG3Q 467892 Ki = 10 nM T17345 C7EJH4 467893 Ki < 2 nM T17345 CL91XC 467894 Ki = 10 nM T17345 CI8A9R 467895 Ki = 6.4 nM T17345 CT9M6G 467896 Ki < 2 nM T17345 C68DYK 467897 Ki = 24 nM T17345 CS8GB6 467898 Ki = 0.1 nM T17345 C3VY2Z 467899 Ki = 0.4 nM T17345 C4WIB5 467900 Ki = 0.1 nM T17345 CI81OG 467901 Ki = 0.2 nM T17345 CL8X1M 467902 Ki = 0.2 nM T17345 CSMT16 467903 Ki = 30 nM T17345 C45HLJ 467904 Ki = 0.4 nM T17345 CRUW28 467905 Ki = 0.1 nM T17345 CF1M8Q 468708 IC50 = 450 nM T17345 CSO8F0 468709 IC50 > 26000 nM T17345 CRP1D3 468710 IC50 > 25000 nM T17345 CQM7K4 468711 IC50 > 15000 nM T17345 CT6B0K 468712 IC50 > 15000 nM T17345 C92GMA 470175 IC50 = 6.1 nM T17345 CS6A3D 470176 IC50 = 2.8 nM T17345 C41BHZ 470177 IC50 = 5.2 nM T17345 C1BU8E 470179 IC50 = 6.7 nM T17345 CA3U5C 470200 IC50 = 3.7 nM T17345 C1Y2GQ 470201 IC50 = 5.9 nM T17345 C4D2QK 470202 IC50 = 6.1 nM T17345 C0V5MT 470264 IC50 = 120 nM T17345 CLY84S 470265 IC50 = 8 nM T17345 CMT51S 470266 IC50 = 44 nM T17345 C76HNV 470281 IC50 = 69 nM T17345 CQA07O 470284 IC50 = 250 nM T17345 CWV91M 470285 IC50 = 19 nM T17345 C25WGL 470286 IC50 = 4.6 nM T17345 CX5KM2 470287 IC50 = 3.2 nM T17345 CPC2W8 470288 IC50 = 4.1 nM T17345 CGI39U 470317 IC50 = 4 nM T17345 CI81MK 470318 IC50 = 850 nM T17345 C3O4TZ 470332 IC50 = 5300 nM T17345 CMJ5I4 470333 IC50 = 1900 nM T17345 CLM7A5 472826 IC50 = 3400 nM T17345 C0IJ7Q 472845 IC50 = 3.8 nM T17345 CM6FH7 472846 IC50 = 6.2 nM T17345 CQGS78 472847 IC50 = 2 nM T17345 C8NJU3 472848 IC50 = 68 nM T17345 CNBY98 472849 IC50 = 14 nM T17345 CIHZ91 472850 IC50 = 33 nM T17345 C9H4YB 472852 IC50 = 277 nM T17345 C7VGW9 472853 IC50 = 20 nM T17345 CVFX53 472910 Ki = 24.4 nM T17345 CERP02 474750 IC50 = 15 nM T17345 C0SG1N 476032 IC50 = 2459 nM T17345 C1Z6AQ 476042 IC50 = 1526 nM T17345 CY37PZ 476043 IC50 = 942 nM T17345 C74WGU 477890 IC50 = 7300 nM T17345 C3JY5Z 479281 IC50 = 700 nM T17345 CM2GT8 479412 IC50 = 76000 nM T17345 CF3C8Q 479413 IC50 = 13000 nM T17345 C41TQB 479416 IC50 = 530 nM T17345 C59FRQ 479418 IC50 = 160000 nM T17345 CF2JD3 479421 IC50 = 6200 nM T17345 CRB65P 481401 IC50 > 19000 nM T17345 COV85S 482165 IC50 = 1300 nM T17345 C9KOB8 485848 IC50 = 0.0021 nM T17345 C3JX2W 490573 IC50 = 5000 nM T17345 C25VUD 490663 Ki = 96.3 nM T17345 CI74ZT 490664 Ki = 4.3 nM T17345 CEW3B0 490665 Ki = 33 nM T17345 C89KLU 490666 Ki = 310 nM T17345 C7LX8H 490667 Ki = 250 nM T17345 CR1SM3 490668 Ki = 49 nM T17345 CLTA76 504022 IC50 = 5000 nM T17345 CN5CJ7 688803 IC50 = 50000 nM T17345 CQ5E7D 789778 Ki = 9.8 nM T17345 C9JQC0 2437106 IC50 = 500 nM T17345 C7RW2A 2731323 Ki = 130 nM T17345 C67UFD 2737412 IC50 = 580 nM T17345 C5F6EO 3010592 IC50 = 6.8 nM T17345 CG6F5S 3132813 Ki = 6.4 nM T17345 C2IFO1 3145500 IC50 = 1900 nM T17345 CFRL82 5183677 IC50 = 830 nM T17345 CHGZ97 5288461 IC50 = 800 nM T17345 CQ1ZH4 5742617 IC50 = 1216 nM T17345 CQ75AN 5742620 IC50 = 624 nM T17345 CT79NS 5742621 IC50 = 1410 nM T17345 CM59DP 5742624 IC50 = 970 nM T17345 C2N0IR 6477203 Ki = 1600 nM T17345 CYP69H 6482470 IC50 = 10000 nM T17345 CXI43R 9805576 IC50 = 1530 nM T17345 CYZ79K 9846618 IC50 = 8.8 nM T17345 CVWX01 9881905 Ki = 15000 nM T17345 CC36EP 9889551 IC50 = 10000 nM T17345 CP75AV 9898639 IC50 = 18000 nM T17345 C5VZN4 9911146 IC50 = 420 nM T17345 C3GI6F 9931657 Ki = 0.005 nM T17345 CL0P6O 9932276 IC50 = 1000 nM T17345 CIDQ05 9952879 Ki = 0.12 nM T17345 CBQK30 9973530 Ki = 4.2 nM T17345 CG9ZU8 9976735 IC50 > 26000 nM T17345 C2C7WX 9980556 Ki = 0.54 nM T17345 C3FR4N 10004772 IC50 = 125 nM T17345 C7RD2X 10007840 Ki = 0.183 nM T17345 C9A1VX 10019413 Ki = 24 nM T17345 CID95L 10030947 Ki = 0.000014 nM T17345 CN4V0B 10053803 Ki = 0.00041 nM T17345 C04LWZ 10060600 Ki = 1.6 nM T17345 CQI0P1 10060703 IC50 = 20 nM T17345 C37ZPO 10065177 Ki = 977.24 nM T17345 C5THD4 10070986 IC50 = 16 nM T17345 C70FRM 10072852 IC50 = 66 nM T17345 CQ8U6T 10090457 Ki > 5000 nM T17345 CSJY78 10246793 Ki = 36 nM T17345 C8ME5O 10260430 IC50 = 2.5 ug.mL-1 T17345 CGT0H9 10326322 Ki = 0.00011 nM T17345 CKFP04 10403719 Ki = 140 nM T17345 C7KXJ2 10404647 IC50 = 560 nM T17345 C9PRM3 10405166 IC50 = 2.8 nM T17345 CTX6H7 10433577 IC50 = 210 nM T17345 CZD4B0 10456691 IC50 = 21000 nM T17345 CB15AR 10457642 IC50 = 1.3 nM T17345 CHM3X4 10478775 Ki = 3400 nM T17345 CPO4W7 10518330 Ki = 9.8 nM T17345 C12BJE 10522269 Ki = 52 nM T17345 CZ8YM9 10544281 Ki = 75 nM T17345 CM95NE 10565157 Ki = 7.1 nM T17345 CLK5H2 10590469 IC50 = 3185 nM T17345 CG83DM 10608757 Ki = 750 nM T17345 C9WCK2 10634047 Ki = 8.6 nM T17345 CI5SU7 10658874 Ki = 10.5 nM T17345 CBXD51 10682649 Ki = 8.8 nM T17345 CXZL07 10709354 Ki = 13 nM T17345 C41ICW 10719122 IC50 = 3100 nM T17345 C0B7YU 10805231 Ki = 131 nM T17345 CHK35G 10807265 Ki = 19 nM T17345 CMF9L1 10826074 Ki = 3.6 nM T17345 C7XFJ5 10828475 Ki = 11 nM T17345 C3R0FI 10860015 IC50 = 10 nM T17345 C0S6TG 10883066 IC50 = 22000 nM T17345 CYWT73 10884015 IC50 = 100000 nM T17345 C9HR0M 10902858 IC50 = 32000 nM T17345 C8B0FL 10961831 IC50 = 5400 nM T17345 C4ZML2 10981577 IC50 = 85 nM T17345 C9D4VK 10991113 IC50 = 44 nM T17345 C9LPA1 10993870 IC50 = 920 nM T17345 CCQ4P6 11003295 IC50 = 2 nM T17345 C2P3AT 11047021 IC50 = 1300 nM T17345 CZ90JL 11058970 IC50 = 450 nM T17345 C4RBD9 11078421 IC50 = 21 nM T17345 CP5YV0 11099765 IC50 = 27000 nM T17345 CY1A7Q 11102571 IC50 = 7 nM T17345 C9ZWB1 11154001 IC50 > 10000 nM T17345 CO2DY5 11247965 Ki = 0.034 nM T17345 C8Q6ZT 11248313 Ki = 2.1 nM T17345 CIG85H 11282247 IC50 = 300 nM T17345 CI2TD8 11340329 IC50 > 10000 nM T17345 C85DMO 11349789 IC50 = 28000 nM T17345 C4EL7T 11430583 IC50 > 10000 nM T17345 CH8IF2 11442040 IC50 > 10000 nM T17345 C41XHB 11452801 IC50 > 10000 nM T17345 CJS58R 11455251 IC50 > 10000 nM T17345 C03JKV 11478803 Ki = 0.0001 nM T17345 C3ROC9 11538533 IC50 < 10 nM T17345 C6K9EH 11573029 IC50 = 630 nM T17345 C1XJI4 11645134 IC50 = 10700 nM T17345 C71ZQD 11645349 IC50 = 34 nM T17345 CYL01H 11651834 IC50 = 9400 nM T17345 CRUQ79 11673839 IC50 = 98000 nM T17345 C8AEX7 11687971 Ki = 500 nM T17345 C19BQV 11688044 IC50 = 8400 nM T17345 CQ4H5E 11744008 IC50 = 9000 nM T17345 CE7DH6 11783065 IC50 = 30000 nM T17345 CTB69W 11822511 IC50 = 47 nM T17345 CR9GN2 11826533 IC50 = 22000 nM T17345 CWP0B9 11846624 IC50 = 1830 nM T17345 CCUF60 11846625 IC50 = 2300 nM T17345 CW5VO2 12214236 Ki = 56000 nM T17345 CU1CF0 12242319 IC50 = 377000 nM T17345 CML17O 12242320 IC50 = 242000 nM T17345 CZO4H8 12242322 IC50 = 57000 nM T17345 C9AQ3V 12242324 IC50 = 740000 nM T17345 C13ZHJ 12517699 IC50 = 28000 nM T17345 CRSM76 12517700 IC50 = 7000 nM T17345 CSN4H6 12517701 IC50 = 8000 nM T17345 CMT96B 12517702 IC50 = 11000 nM T17345 C32RLQ 12517703 IC50 = 903000 nM T17345 C3G8JV 12517705 IC50 = 168000 nM T17345 CYPT41 12655201 IC50 = 370 nM T17345 CI0Y1T 12655204 IC50 = 58 nM T17345 CUXC87 12803287 IC50 = 340000 nM T17345 C98JXK 13112734 IC50 = 120 nM T17345 CX3Q6D 13112736 IC50 = 49 nM T17345 C8EIC5 13112740 IC50 = 29 nM T17345 C1INA2 13112752 IC50 = 310 nM T17345 C5X3WZ 13112757 IC50 = 44 nM T17345 C84HXC 13170795 IC50 = 14000 nM T17345 CU4O5B 13739857 IC50 = 61 nM T17345 CZLB08 13877973 IC50 = 230 nM T17345 CU8A4L 13877981 IC50 = 1110 nM T17345 CZV23T 13953684 IC50 = 67 nM T17345 CIW97R 13953685 IC50 = 93 nM T17345 CQFS01 13953687 IC50 = 110 nM T17345 C49DCF 13953688 IC50 = 170 nM T17345 C47HUP 13953689 IC50 = 20 nM T17345 C25SRU 13989362 IC50 = 5.3 nM T17345 CHI71Y 13989363 IC50 = 5.4 nM T17345 CRN23J 14083105 IC50 = 72 nM T17345 CS1G8K 14503206 IC50 = 40 nM T17345 CD84TM 14503207 IC50 = 70 nM T17345 CZET95 14560097 IC50 = 3 nM T17345 CAM5O1 14570150 Ki = 0.8 nM T17345 C8XLI9 14570153 IC50 = 66 nM T17345 CM49FY 14570156 IC50 = 110 nM T17345 C46HSO 14570159 IC50 = 14 nM T17345 CEL4B9 14570163 IC50 = 46 nM T17345 C6N4JB 14570319 IC50 = 300 nM T17345 C20TUW 14570320 IC50 = 630 nM T17345 CFQ37R 14570325 IC50 = 1800 nM T17345 CK5JI7 14570338 IC50 = 540 nM T17345 C3B7AQ 14570339 IC50 = 140 nM T17345 C9W4IP 14776576 IC50 = 6.4 nM T17345 C9V3SY 14776579 IC50 = 88 nM T17345 CX4U2T 14776583 IC50 = 57 nM T17345 CU1M4X 14776589 IC50 = 5.3 nM T17345 CWDB20 14776590 IC50 = 5.9 nM T17345 C9EW5Z 14776615 IC50 = 6000 nM T17345 CA4HC9 14776619 IC50 > 20000 nM T17345 CW5C6T 14801655 IC50 = 32 nM T17345 CBKR63 14801660 IC50 = 35 nM T17345 C68YXF 14801666 IC50 = 30 nM T17345 C4UVQ0 14840934 IC50 = 27000 nM T17345 CL5H0X 14840943 IC50 = 35 nM T17345 CORH59 14840958 IC50 = 50 nM T17345 C7VK0C 15021215 IC50 = 1.34 nM T17345 C4D8IR 15523786 Ki = 14.1 nM T17345 CW1QA4 15523787 Ki = 0.107 nM T17345 C6QM7Z 15616236 IC50 = 19000 nM T17345 C8W1DB 15616238 IC50 > 50000 nM T17345 CQ1TU0 16038397 Ki = 9.6 nM T17345 CWKX69 16086910 Ki = 110000 nM T17345 C6V7GN 16086911 Ki = 35000 nM T17345 C3X9DE 16086912 Ki = 3900 nM T17345 C9KZ4H 16086913 Ki = 33000 nM T17345 CTK25X 16086914 Ki = 69000 nM T17345 C7MA5T 16086915 Ki = 13000 nM T17345 CD59VR 16086916 Ki = 35000 nM T17345 C6UX1P 16086917 Ki = 109000 nM T17345 CRWB95 16086918 Ki = 13000 nM T17345 C0RE7Z 16086919 Ki = 12000 nM T17345 C1BYA7 16110323 IC50 = 1460 nM T17345 C4XBM2 16110326 IC50 = 1380 nM T17345 CB36UF 16110328 IC50 = 5710 nM T17345 CS9FR8 16110329 IC50 = 1160 nM T17345 C31SJW 16110337 IC50 = 400 nM T17345 CJ73WY 16110338 IC50 = 1460 nM T17345 C3LHA7 16110339 IC50 = 14300 nM T17345 C8OYD1 16110341 IC50 = 1220 nM T17345 C81MTW 16110344 IC50 = 1380 nM T17345 CZJM43 16732891 IC50 = 2900 nM T17345 CGM38B 16732892 IC50 = 6000 nM T17345 CMC21Z 16732893 IC50 = 5800 nM T17345 C9IG0J 16733029 IC50 = 2700 nM T17345 CHL6F9 16733030 IC50 > 31000 nM T17345 C8X9EC 16733031 IC50 > 31000 nM T17345 CW5SB7 16733033 IC50 > 28000 nM T17345 CM80YI 16733034 IC50 = 5800 nM T17345 CM1I4D 16733035 IC50 > 32000 nM T17345 CP8VS3 16733036 IC50 = 1400 nM T17345 C83VHB 16733162 IC50 = 1400 nM T17345 CED2R5 16733163 IC50 = 2900 nM T17345 CDA8P5 16733164 IC50 = 18000 nM T17345 CXA71B 16733165 IC50 = 32000 nM T17345 CC09RL 19089924 IC50 = 430 nM T17345 CK1P0V 21496446 IC50 = 140 nM T17345 C7B8CR 21705470 IC50 = 83300 nM T17345 C27WPQ 23161237 IC50 = 1100 nM T17345 CE2XM5 23629645 Ki = 800 nM T17345 CT2G9I 23647976 IC50 = 2100 nM T17345 CUSF67 23648073 Ki = 94000 nM T17345 CI2F9K 23648074 Ki = 28000 nM T17345 C4SXQ7 23648075 Ki = 15000 nM T17345 CDUX91 23648076 Ki = 9500 nM T17345 CE4G3V 23729147 IC50 > 125000 nM T17345 C7TLP1 24202945 Ki = 2000 nM T17345 C4S9RX 24202946 Ki = 8000 nM T17345 C6H1RM 24202947 Ki = 8000 nM T17345 C7AXQ6 24203165 Ki = 6000 nM T17345 CUC7I6 24203167 Ki = 4000 nM T17345 CG7RU5 24203941 Ki = 3000 nM T17345 C9BO1H 24203942 Ki = 5000 nM T17345 COCG69 24203943 Ki = 3000 nM T17345 C6S0FC 24204135 Ki = 5000 nM T17345 C2M1JB 24204136 Ki = 11000 nM T17345 C5S8PW 24204221 Ki = 4000 nM T17345 C63PUM 24204222 Ki = 3000 nM T17345 C89JMH 24204223 Ki = 5000 nM T17345 CN13ZR 24204418 Ki = 5000 nM T17345 C1IN2K 24204433 Ki = 3000 nM T17345 C6Y0ZX 24204434 Ki = 7000 nM T17345 CP73JD 24204806 Ki = 5000 nM T17345 C6M5YP 24204807 Ki = 8000 nM T17345 CA3BT0 24204808 Ki = 4000 nM T17345 CEK8R6 24777136 IC50 = 39 nM T17345 C6O5CL 24778299 IC50 = 25 nM T17345 CL7KN4 24950538 IC50 = 2600 nM T17345 C2C4FZ 24950539 IC50 = 3000 nM T17345 C9LY5G 24950540 IC50 = 33000 nM T17345 CPEF92 24950541 IC50 > 30000 nM T17345 CD8QM2 24950542 IC50 = 28000 nM T17345 CX5Q0K 24950543 IC50 > 26000 nM T17345 CH9A4V 24950693 IC50 > 29000 nM T17345 CG6A8V 24950694 IC50 > 15000 nM T17345 C6F2CR 24950695 IC50 > 26000 nM T17345 CX1AR8 24950696 IC50 > 30000 nM T17345 C1PHA0 24950697 IC50 = 16000 nM T17345 CG2B8O 24950698 IC50 = 30000 nM T17345 CX97IY 24950699 IC50 > 28000 nM T17345 C32OJF 24950851 IC50 = 27000 nM T17345 CCY8U4 24950852 IC50 > 29000 nM T17345 C17DAP 24950853 IC50 > 29000 nM T17345 CPDN34 24950854 IC50 > 27000 nM T17345 C2BXV5 25002412 IC50 > 125000 nM T17345 CQ3AV2 25002763 IC50 > 125000 nM T17345 CNBS61 25007427 IC50 = 55200 nM T17345 C1ER2L 25007788 IC50 > 125000 nM T17345 CIB13V 25058133 IC50 = 1280 nM T17345 CZ9L1Y 25093361 IC50 = 1700 nM T17345 COHL97 25093362 IC50 = 1360 nM T17345 C7PUO6 25093363 IC50 = 1250 nM T17345 CZE0Q4 25093364 IC50 = 7200 nM T17345 CGRF64 25093365 IC50 = 1420 nM T17345 CU0M5T 25093366 IC50 = 2770 nM T17345 CMQR72 25093367 IC50 = 3370 nM T17345 COE57Z 25093368 IC50 = 4200 nM T17345 CJV6X5 25093369 IC50 = 1360 nM T17345 C49FRJ 25093370 IC50 = 1380 nM T17345 C6W1TN 25107577 IC50 = 3500 nM T17345 CHU9G1 25107640 IC50 = 1500 nM T17345 C5WV3Q 25107642 IC50 = 5600 nM T17345 C2FU7W 25107643 IC50 = 2500 nM T17345 C5EP2L 25107644 IC50 = 2800 nM T17345 C3YT9V 25107645 IC50 = 2900 nM T17345 CQV0S4 25107646 IC50 = 2600 nM T17345 CO01BE 25138222 IC50 = 3200 nM T17345 CCK4R2 25138223 IC50 = 1300 nM T17345 C7P2RD 25138224 IC50 = 1180 nM T17345 C4VFL0 25138225 IC50 = 57 nM T17345 CR2MW1 25138226 IC50 = 130 nM T17345 CQO1Y3 25138227 IC50 = 360 nM T17345 COB9G8 25181586 IC50 > 33000 nM T17345 CF8EX5 25187895 IC50 = 200 nM T17345 C5BH0D 25187896 IC50 = 290 nM T17345 C3F5HV 25187897 IC50 = 210 nM T17345 CJ51SH 25187898 IC50 = 180 nM T17345 C1J4CH 25195124 IC50 = 750 nM T17345 C4P5UX 25195125 IC50 = 1410 nM T17345 C8IJB9 25218207 IC50 > 31000 nM T17345 C2SY4Z 25243853 Ki = 10000 nM T17345 CS6HE5 42627761 IC50 = 110000 nM T17345 C3C2GH 44123767 IC50 = 2370 nM T17345 C93GYN 44123768 IC50 = 2150 nM T17345 COI2S4 44136999 Ki = 15430 nM T17345 CWH0S1 44137255 Ki = 590 nM T17345 CI0BF4 44201386 IC50 = 19 nM T17345 CZ6DE0 44221143 IC50 = 300 nM T17345 CL8B5Q 44221144 IC50 = 840 nM T17345 CSJ28V 44221145 IC50 = 280 nM T17345 COT01Q 44221146 IC50 = 620 nM T17345 CS14YU 44221147 IC50 = 300 nM T17345 CA64NZ 44221340 IC50 = 600 nM T17345 CK5OL1 44221343 IC50 = 2600 nM T17345 CW0IM7 44221344 IC50 = 260 nM T17345 C0QZ7V 44221345 IC50 = 290 nM T17345 C74PHB 44221346 IC50 = 2200 nM T17345 CW39YO 44221347 IC50 = 350 nM T17345 CBHT60 44221538 IC50 = 260 nM T17345 CN5QV6 44221539 IC50 = 540 nM T17345 C9O1JI 44239402 IC50 = 173 nM T17345 CL13YN 44239406 IC50 = 19.9 nM T17345 C2PA5U 44239552 IC50 = 1790 nM T17345 C4NWP5 44246325 Ki = 2500 nM T17345 C2EW0I 44246326 Ki = 770 nM T17345 CSD8T0 44246327 Ki = 650 nM T17345 CMKF08 44246328 Ki = 12000 nM T17345 CAO87V 44246329 Ki = 5300 nM T17345 CLU2V3 44246330 Ki = 4600 nM T17345 CZ8U9G 44264907 IC50 = 1 nM T17345 CCJ0E5 44272288 IC50 = 27 nM T17345 CZ83VS 44273520 Ki = 776.25 nM T17345 CB9ZO8 44281305 IC50 = 320 nM T17345 C2O1KM 44281312 IC50 = 650 nM T17345 CFB79E 44282924 Ki = 46.2 nM T17345 C8QZ2E 44282925 Ki = 55.7 nM T17345 C51OKF 44282953 Ki = 0.131 nM T17345 C41RVE 44283340 IC50 = 1.5 nM T17345 CTZ9E5 44291963 Ki = 0.00033 nM T17345 C0D1VX 44291964 Ki = 0.0006 nM T17345 CHSF50 44291965 Ki = 0.00035 nM T17345 CDW63J 44292014 Ki = 0.00062 nM T17345 CG4KS0 44292015 Ki = 0.00021 nM T17345 C2DQ9E 44300934 IC50 = 1000 nM T17345 CN9U6W 44300964 IC50 = 420 nM T17345 CEV8X6 44300967 IC50 = 220 nM T17345 C54FJZ 44301716 IC50 = 190 nM T17345 C9JG5P 44308541 IC50 = 4.6 nM T17345 C0LZ8X 44308557 IC50 = 5.7 nM T17345 C7Q4RC 44309078 IC50 = 10.2 nM T17345 C8KST2 44314297 IC50 = 12 nM T17345 CBK5E3 44338827 IC50 = 14 nM T17345 CE14LA 44342970 IC50 = 27 nM T17345 CV6U1R 44343198 IC50 = 600 nM T17345 C6GME8 44346127 IC50 = 200 nM T17345 CN0GE5 44366301 Ki = 0.00019 nM T17345 C05HEV 44366644 IC50 = 18 nM T17345 C8AQ0F 44372902 IC50 = 0.84 nM T17345 C5F0ZB 44378252 Ki = 0.29 nM T17345 CZ7Y4L 44378321 Ki = 9.87 nM T17345 C3W2YH 44378322 Ki = 0.69 nM T17345 CM4Z7A 44421498 Ki = 0.077 nM T17345 CZ4CF9 44424991 IC50 = 2800 nM T17345 C0G4XZ 44523554 IC50 = 382.1 nM T17345 CB3D5L 44529842 IC50 > 100000 nM T17345 CPDY84 44531062 IC50 = 7.6 nM T17345 CN76FA 44568860 IC50 = 20 nM T17345 CPT49L 44582168 IC50 = 560 nM T17345 C0O4GX 44582169 IC50 = 1408 nM T17345 CM67QY 44582180 IC50 = 9340 nM T17345 CPS34N 44654525 IC50 = 2900 nM T17345 CMH39V 45267084 IC50 > 22000 nM T17345 C2V1MK 45267934 IC50 = 110000 nM T17345 CA53OY 45267939 IC50 > 27000 nM T17345 CYGI67 45268817 IC50 > 16000 nM T17345 C9H3DZ 45269661 IC50 > 20000 nM T17345 CE6W3J 45269665 IC50 > 24000 nM T17345 CW82HJ 45270497 IC50 > 28000 nM T17345 CW37YT 45270501 IC50 > 19000 nM T17345 CUNA34 45270504 IC50 > 21000 nM T17345 CGU1K7 45271328 IC50 > 25000 nM T17345 C17OKU 45271331 IC50 > 19000 nM T17345 C9M2ET 45271332 IC50 > 22000 nM T17345 CVGQ38 45272213 IC50 = 813000 nM T17345 CTFO90 45273072 IC50 > 23000 nM T17345 C50PYG 45273073 IC50 > 42000 nM T17345 C70SNR 45481871 IC50 = 1200 nM T17345 CM65ZU 45481878 IC50 = 60 nM T17345 CIGZ82 45481879 IC50 = 2300 nM T17345 CM3BD5 45481892 IC50 = 290 nM T17345 CP82LD 45481893 IC50 = 1580 nM T17345 CD1G7Q 45481939 IC50 = 400 nM T17345 CM1BK5 45481950 IC50 = 88 nM T17345 C1YAE7 46231368 IC50 = 4000 nM T17345 C1PJ2K 46231369 IC50 > 200000 nM T17345 CV38CS 46231370 IC50 > 200000 nM T17345 C5WM1J 46231371 IC50 > 200000 nM T17345 C5D7UV 46231372 IC50 > 200000 nM T17345 C9OER4 46231373 IC50 > 200000 nM T17345 CW0UO4 46231409 IC50 > 200000 nM T17345 C7OG0U 46231410 IC50 > 200000 nM T17345 CU5T7G 46231411 IC50 > 200000 nM T17345 COML63 46231412 IC50 > 200000 nM T17345 CK21OD 46231413 IC50 > 200000 nM T17345 C7Y5MX 46231414 IC50 > 200000 nM T17345 CN3HM6 46844539 Ki = 49.8 nM T17345 C5NOF1 46844540 Ki = 11.8 nM T17345 C9OM6V 46844541 Ki = 13 nM T17345 C2K9SC 46844649 Ki = 188 nM T17345 C6N1YZ 46861681 IC50 = 900 nM T17345 CY3M7K 46861682 IC50 = 1000 nM T17345 CIL1Z3 46886064 IC50 = 2000 nM T17345 CDV7P4 46886065 IC50 = 500 nM T17345 CO6E2M 46886122 IC50 = 500 nM T17345 CVX23N 46886123 IC50 = 800 nM T17345 CE9TL8 46886124 IC50 = 1000 nM T17345 COQ64I 46886125 IC50 = 1000 nM T17345 CPF1G2 46886145 IC50 = 2000 nM T17345 CB4YL0 46886146 IC50 = 2000 nM T17345 CM8B7K 46886147 IC50 = 800 nM T17345 C42TQK 46886148 IC50 = 3000 nM T17345 C5USK9 46886149 IC50 = 700 nM T17345 CCGH29 46886469 IC50 = 4000 nM T17345 C3PZL9 46886489 IC50 = 1000 nM T17345 CF27TO 46886490 IC50 = 3000 nM T17345 C26DLM 46886513 IC50 = 6000 nM T17345 CN4JM7 46886546 IC50 = 3000 nM T17345 CLY37J 46898100 Ki = 34 nM T17345 CQ3E4W 46898103 Ki = 7.6 nM T17345 C9H4WN 46905455 Ki = 9 nM T17345 CF4UK7 46907163 Ki = 24.5 nM T17345 CL14GQ 50992060 Ki = 22.5 nM T17345 CE0VL8 50994805 IC50 = 300000 nM T17345 CJA45X 52914860 IC50 = 90 nM T17345 CV21AI 52914861 IC50 = 100 nM T17345 CT8R2P 52918390 Ki = 1026 nM T17345 C7BY6M 52942956 Ki = 830 nM T17345 CE02NU 52943039 IC50 = 42000 nM T17345 CX24TS 52943277 IC50 = 340 nM T17345 CA62KU 52944152 Ki = 1600 nM T17345 CE37DL 52944456 IC50 = 314 nM T17345 CQV34K 52945403 Ki = 1100 nM T17345 C97XZA 52946619 Ki = 11000 nM T17345 CD9S4I 52947801 Ki = 4300 nM T17345 CA6IL3 52947802 Ki = 1300 nM T17345 C0MQ9Y 53346505 Ki = 1138 nM T17345 C2EGS5 53346506 Ki = 12.2 nM T17345 CAK50X 53346507 Ki = 26.3 nM T17345 COSG28 53346508 Ki = 12 nM T17345 C5U3KJ 53346509 Ki = 11.1 nM T17345 CD60FA 53346510 Ki = 5.8 nM T17345 CX2NV9 53346511 Ki = 4.5 nM T17345 CK72UF 53387838 IC50 > 100000 nM T17345 CXOL35 56595784 Ki = 572 nM T17345 CT45OM 56595785 Ki = 854 nM T17345 C9OW8X 56658455 IC50 > 100000 nM T17345 C1VYN7 56658457 IC50 > 100000 nM T17345 CDWN05 56658459 IC50 > 100000 nM T17345 CEX01L 56659280 Ki = 323 nM T17345 C6UHW8 56659281 Ki = 11.1 nM T17345 C0OSM1 56662749 Ki = 95.6 nM T17345 CO14BL 56665108 IC50 = 155 nM T17345 C6ER2F 56665410 IC50 > 100000 nM T17345 C1KWA9 56665412 IC50 > 100000 nM T17345 C7IX2A 56665414 IC50 > 100000 nM T17345 CPO4V8 56665416 IC50 > 100000 nM T17345 CUPO65 56666113 IC50 > 20000 nM T17345 CDC24L 56666218 Ki = 44.1 nM T17345 C9C7KW 56666219 Ki = 85 nM T17345 CH91WP 56666648 IC50 = 14000 nM T17345 CMHP59 56668551 IC50 = 5330 nM T17345 CQP5U2 56668841 IC50 > 100000 nM T17345 C2F0BA 56668843 IC50 > 100000 nM T17345 CDGX83 56668845 IC50 > 100000 nM T17345 CML5O9 56669623 Ki = 743 nM T17345 C2FBW1 56669624 Ki = 702 nM T17345 CCS0D3 56669625 Ki = 253 nM T17345 CP91XV 56673137 Ki = 20.9 nM T17345 C3JKO4 56673138 Ki = 22.2 nM T17345 COK3Z5 56675436 IC50 = 134 nM T17345 CUQ67O 56675715 IC50 > 100000 nM T17345 C6RCQ7 56676341 IC50 > 20000 nM T17345 C8AQ1O 56676459 Ki = 138 nM T17345 C7T2IG 56676460 Ki = 27.5 nM T17345 COA13E 56676461 Ki = 245 nM T17345 COG17M 56678776 IC50 = 548 nM T17345 C6VS9Y 56679010 IC50 = 21800 nM T17345 CJZ9B0 56679012 IC50 > 100000 nM T17345 C2B0OZ 56679014 IC50 > 100000 nM T17345 C90TMJ 56679774 Ki = 129 nM T17345 C29UVR 56679775 Ki = 10.1 nM T17345 COF0V7 56680536 IC50 = 49.04 nM T17345 CKX0H5 56682332 IC50 > 100000 nM T17345 CLGR37 56682334 IC50 > 100000 nM T17345 CDH01Q 56683111 Ki = 41.1 nM T17345 CRLK58 57381314 IC50 = 289 nM T17345 CZBG69 57381532 IC50 = 599 nM T17345 CRB3F1 57404325 IC50 > 250000 nM T17345 CA6DB4 57404326 IC50 = 50000 nM T17345 CBOX49 59608000 Ki = 4330 nM T17345 CTW7K2 60142113 IC50 = 5960 nM T17345 C7NCS0 60142250 IC50 = 2110 nM T17345 CC1X7M 60142382 IC50 = 1610 nM T17345 C3SH4V 60194459 Ki = 33.6 nM T17345 C25XOP 60199138 Ki = 18.1 nM T17345 C0WYU6 60199139 Ki = 20.2 nM T17345 CSA7P4 66563689 Ki = 47.6 nM T17345 CLJ4S9 66924089 IC50 = 15000 nM T17345 C47NRM 67607115 Ki = 1164 nM T17345 C5C0VZ 67607544 Ki = 1086 nM T17345 C8YM7S 67607902 Ki = 663 nM T17345 CVQW83 67615348 Ki = 320 nM T17345 C23NBA 67889361 Ki = 943 nM T17345 C95DAH 67889364 Ki = 2.9 nM T17345 CG5J2I 70687448 IC50 > 250000 nM T17345 CJAF56 70689505 IC50 > 250000 nM T17345 CZ48NJ 70695829 IC50 = 340 nM T17345 C0OB8G 71307952 IC50 = 57 nM T17345 C7KSO5 71449539 IC50 = 420 nM T17345 CJ6SQ8 71451328 IC50 = 33 nM T17345 CQ5YE6 71451881 Ki = 4680 nM T17345 C2F5XK 71453144 IC50 = 800 nM T17345 CTP47E 71454881 IC50 = 1070 nM T17345 CB1WD6 71456658 IC50 = 32 nM T17345 CSU17Q 71460350 IC50 = 18 nM T17345 C0UXW2 71462049 IC50 = 33 nM T17345 C7FEJ4 71462050 IC50 > 100000 nM T17345 CFP1O3 71463580 IC50 = 150 nM T17345 CKA6Q2 71463581 Ki = 11 nM T17345 C9SU7T 71520360 Ki > 55000 nM T17345 C9M2JK 71520483 Ki > 332000 nM T17345 C5N4XG 71521660 Ki > 110000 nM T17345 CGP9N4 71525312 IC50 = 1300 nM T17345 C3GN0W 71560185 IC50 = 400 nM T17345 CRZK12 71560290 IC50 = 250 nM T17345 CF06NE 71560291 IC50 = 1500 nM T17345 C2SJ7K 71560296 IC50 = 60 nM T17345 CCP40I 71560419 IC50 = 45 nM T17345 CR38HE 71560424 IC50 = 140 nM T17345 C06WSC 71560425 IC50 = 260 nM T17345 CV3A1O 71680871 IC50 = 190 nM T17345 CL5G6W 71680872 IC50 = 3650 nM T17345 CN8E7Q 71680873 IC50 = 250 nM T17345 CLT08Y 71680874 IC50 = 1000 nM T17345 CBW3F2 71680875 IC50 = 3900 nM T17345 CX82PD 71680876 IC50 = 2100 nM T17345 CGR6J5 71680877 IC50 = 5900 nM T17345 C23EQL 71681031 IC50 = 2200 nM T17345 CI9Y4J 71681032 IC50 = 7200 nM T17345 CO4V1J 71681033 IC50 = 2100 nM T17345 CU5IC1 71681034 IC50 = 450 nM T17345 C3I5KR 71681035 IC50 = 3100 nM T17345 CYG8K1 71681036 IC50 = 12 nM T17345 CNT81J 71681037 IC50 = 14 nM T17345 CCS0L2 71681187 IC50 = 4.7 nM T17345 C1X8KC 71681188 IC50 = 4.6 nM T17345 C46UPB 71681189 IC50 = 32 nM T17345 C7A1WK 71681190 IC50 = 340 nM T17345 CTIX90 71681191 IC50 = 5.6 nM T17345 C38MXU 71681192 IC50 = 46 nM T17345 CMJ47I 72771095 Ki = 1101 nM T17345 CZ4D3T 73386686 IC50 = 180 nM T17345 C8HKV5 76308482 IC50 = 3000 nM T17345 CR1SA3 76310814 Ki = 4000 nM T17345 CBH3C5 76311133 Ki = 841 nM T17345 CE8K7X 76314747 Ki > 5000 nM T17345 CWYV16 76314759 Ki = 1607 nM T17345 C9L4RE 76314760 Ki = 2922 nM T17345 CWN21Q 76318014 Ki = 4000 nM T17345 CE9Q3J 76318015 Ki = 200 nM T17345 CFM0V3 76318330 Ki = 749 nM T17345 CY8T3V 76319350 IC50 = 1.3 nM T17345 C17BXW 76319351 IC50 = 8.9 nM T17345 C0WMC2 76319379 IC50 = 10 nM T17345 C1B0TE 76322025 Ki = 723 nM T17345 C7N0YG 76323015 IC50 = 7300 nM T17345 CN7LS9 76325171 IC50 = 100 nM T17345 CL62UB 76325172 IC50 = 500 nM T17345 C2TF7J 76325354 Ki = 6000 nM T17345 CZ5DA3 76325652 Ki > 3000 nM T17345 C3PJ8X 76325653 Ki > 3000 nM T17345 CUC0O5 76325779 IC50 > 1000000 nM T17345 CQYO16 76328899 Ki = 3000 nM T17345 C12PIT 76328900 Ki = 3000 nM T17345 C1W8SP 76329213 Ki = 610 nM T17345 CVS27U 76329214 Ki = 437 nM T17345 CU1N3X 76330211 IC50 = 94 nM T17345 C8CQ5G 76332587 Ki = 3000 nM T17345 CM7X0D 76332864 Ki = 1564 nM T17345 CIAJ89 76336478 Ki = 2299 nM T17345 CYZJ97 76336479 Ki > 5000 nM T17345 C60IHU 76336487 Ki = 170 nM T17345 CJEA39 77461251 IC50 = 1200 nM T17345 CI0BY7 86276188 IC50 = 688 nM T17345 CLN0B2 86276189 IC50 = 625 nM T17345 CMF27J 86577836 IC50 = 172 nM T17345 C9EMA6 86577876 IC50 = 127 nM T17345 CC0F4M 86577948 IC50 = 136 nM T17345 CMV52E 86578029 IC50 = 208 nM T17345 C6F0NA 86578120 IC50 = 477 nM T17345 CUMG18 86578123 IC50 = 170 nM T17345 C4L6CM 86578162 IC50 = 49 nM T17345 C7T4CU 86578197 IC50 = 147 nM T17345 C37MOB 86578230 IC50 = 148 nM T17345 CQ3I8M 86578301 IC50 = 174 nM T17345 CVD2Y7 90666046 IC50 = 2730 nM T17345 CQS9A6 90666047 IC50 = 3100 nM T17345 C1UY6B 90666049 IC50 = 8720 nM T17345 CIG5W1 121493974 Ki = 200.77 nM T17345 CY21HZ 122164615 IC50 = 92 nM T17345 C8QB7N 124080837 IC50 = 511 nM T17345 C9NQ7B 124080838 IC50 = 1372 nM T17345 CW2D6Y 124081250 Ki = 388.62 nM T17345 CS04TC 124081251 Ki = 234.23 nM T17345 CO5MJ2 124220265 IC50 = 45 nM T17345 CE5F7Z 124220266 IC50 = 16 nM T17345 C6WU1A 124220267 IC50 = 41 nM T17345 CRE75U 127031638 IC50 = 30000 nM T17345 CY2W5J 127032512 IC50 > 100000 nM T17345 CCQ0D9 127032513 IC50 = 56400 nM T17345 CJ2Q3G 127032813 IC50 = 2400 nM T17345 CAVH35 127033390 Ki = 5.83 nM T17345 C2J9OY 127033391 IC50 = 700 nM T17345 CWK31L 127033392 IC50 = 300 nM T17345 CO9HL0 127033684 IC50 = 8000 nM T17345 C3HRW8 127033994 IC50 > 100000 nM T17345 CBT27N 127034482 IC50 = 5000 nM T17345 CT2OP4 127034483 IC50 = 7000 nM T17345 C6V8HZ 127034484 IC50 = 20000 nM T17345 CK7AG3 127036397 IC50 = 42000 nM T17345 CU7ZS5 127041310 IC50 = 310 nM T17345 C6ZX0J 127041311 IC50 = 310 nM T17345 C2WOC5 127041312 IC50 = 110 nM T17345 C8FD5L 127041909 IC50 = 2 nM T17345 C5Q2OX 127041910 IC50 = 42400 nM T17345 CD8MQ0 127041911 IC50 = 720 nM T17345 C2ILO0 127041912 IC50 = 320 nM T17345 COL16A 127043134 Ki = 2494.9 nM T17345 CWQ6Y4 127043135 Ki = 346.15 nM T17345 CE2R6W 127043324 Ki = 158.77 nM T17345 CEM63B 127043325 Ki = 376.62 nM T17345 C6BF8K 127045460 Ki = 451.15 nM T17345 C14WFB 129906767 IC50 = 72490 nM T17345 CEWR32 130301107 IC50 = 935 nM T17345 CM7E0A 132574708 IC50 = 52000 nM T17345 C4W5JI 134132161 IC50 = 2500 nM T17345 C32OQG 134133398 IC50 > 10000 nM T17345 C4W7YT 134135190 IC50 = 920 nM T17345 CW84JC 134135508 IC50 = 33.56 nM T17345 CF2T9N 134136051 IC50 > 10000 nM T17345 CI45FO 134136319 IC50 = 36.01 nM T17345 C17NRB 134136557 IC50 > 10000 nM T17345 CW0P8B 134136864 IC50 = 32.49 nM T17345 CS27VL 134138165 IC50 = 7.46 nM T17345 CP5IW7 134138953 IC50 = 9200 nM T17345 CCWD64 134139368 IC50 = 1100 nM T17345 CVZI26 134141070 IC50 = 86.11 nM T17345 CTO84X 134141850 IC50 > 10000 nM T17345 C34GRK 134142208 IC50 = 11.07 nM T17345 C3WXJ9 134143008 IC50 = 2100 nM T17345 CWT7F2 134144326 IC50 = 760 nM T17345 CY1X2T 134144992 IC50 = 6.46 nM T17345 C20VFD 134145574 IC50 = 4.08 nM T17345 C86PJW 134146078 IC50 > 10000 nM T17345 C1KFQ9 134147493 IC50 > 10000 nM T17345 CTHA87 134147818 IC50 = 18.28 nM T17345 CQG73J 134147949 IC50 > 10000 nM T17345 CCZ38F 134148801 IC50 > 10000 nM T17345 C2H7AI 134149549 IC50 = 4200 nM T17345 CQ0B2P 134150774 IC50 = 8.23 nM T17345 CA0J6U 134151081 IC50 = 56.75 nM T17345 C3RTP9 134152596 IC50 > 10000 nM T17345 CL72SR 134153211 IC50 > 10000 nM T17345 C2B4RW 134154165 IC50 = 3.72 nM T17345 CK6CQ1 134154523 IC50 > 75000 nM T17345 C18MPZ 134154991 IC50 = 46.62 nM T17345 C5MA8G 134155232 IC50 > 10000 nM T17345 C31ZAM 134156833 IC50 = 2800 nM T17345 C1IX4T 134812633 IC50 = 308 nM T17345 C0LJE4 134816733 IC50 = 11990 nM T17345 C4SZU6 134816735 IC50 = 15320 nM T17345 C3MKJ4 134816970 IC50 = 3670 nM T17345 CCT84X 135399760 IC50 > 240000 nM T17345 CQ4F8Y 135402053 IC50 = 910 nM T17345 C6AY2U 135403832 IC50 > 20000 nM T17345 C0LTC1 135404992 IC50 = 2100 nM T17345 C9EA3J 135407589 IC50 > 100000 nM T17345 C3MHI2 135427303 IC50 = 640 nM T17345 CSNH87 135431649 IC50 = 2100 nM T17345 CJ51DM 135443603 IC50 = 83 nM T17345 CS0I8R 135469335 IC50 > 95000 nM T17345 CS4M7U 135471854 IC50 = 170 nM T17345 C7YPI6 135481470 IC50 = 330 nM T17345 C7BQ1O 135487985 IC50 = 420 nM T17345 C79OVQ 135488791 IC50 = 11 nM T17345 CPZ72B 135488819 IC50 = 460 nM T17345 C5WV3M 135488820 IC50 = 110 nM T17345 CD40CJ 135502983 IC50 > 26000 nM T17345 C98GZD 135511915 IC50 > 54000 nM T17345 CFH82R 135516724 IC50 > 32000 nM T17345 CLB45I 135543610 IC50 > 62000 nM T17345 CK4FS8 135543796 IC50 = 7000 nM T17345 CV7HQ6 135545795 IC50 = 10000 nM T17345 C8N5QD 135545810 IC50 > 21000 nM T17345 CCF8H5 135545819 IC50 > 80000 nM T17345 C9K8DE 135545856 IC50 = 11000 nM T17345 C9Z4ES 135567027 IC50 > 20000 nM T17345 CE5O9J 135570463 IC50 = 22600 nM T17345 C06IDH 135746097 IC50 > 30000 nM T17345 CGLI18 135749904 IC50 = 120 nM T17345 CQ49YZ 135749905 IC50 > 39000 nM T17345 CBUS79 135749906 IC50 > 37000 nM T17345 C2HZK8 135749907 IC50 > 37000 nM T17345 CD48XU 135749908 IC50 > 35000 nM T17345 C9NZA4 135749909 IC50 > 35000 nM T17345 C0ME1H 135749910 IC50 = 33000 nM T17345 CMVH39 135749911 IC50 > 35000 nM T17345 CR4DU1 135749912 IC50 > 35000 nM T17345 C1H6ZF 135749913 IC50 > 31000 nM T17345 CR5NK7 135749914 IC50 > 24000 nM T17345 C1LV7B 135749915 IC50 > 32000 nM T17345 CQF8P5 135800109 IC50 > 24000 nM T17345 C4IDQ3 135855753 IC50 = 66600 nM T17345 C39FIY 135855754 IC50 = 20300 nM T17345 C0N1LQ 135855759 IC50 = 66600 nM T17345 C6A4QR 135855760 IC50 = 100000 nM T17345 CRV4K7 135855761 IC50 = 10200 nM T17345 CAUV24 135855764 IC50 = 72600 nM T17345 CYAS86 135855765 IC50 = 37300 nM T17345 CTG51U 135887103 IC50 = 4700 nM T17345 CE6TP5 135887104 IC50 = 8500 nM T17345 CY5H4A 135887105 IC50 = 400 nM T17345 CHT2O4 135887106 IC50 = 220000 nM T17345 CWL71S 135887124 IC50 = 2000 nM T17345 CNKW46 135887125 IC50 = 12000 nM T17345 CH1W2S 135887126 IC50 = 210 nM T17345 C6U0PF 135887127 IC50 = 250 nM T17345 COA6S0 135887128 IC50 = 1950 nM T17345 CBO9A7 135887129 IC50 = 320 nM T17345 CFIG79 135887147 IC50 > 1000000 nM T17345 CDA05G 135887148 IC50 > 1000000 nM T17345 CZB8O6 135960753 IC50 = 22000 nM T17345 CZ6C4R 135964391 IC50 > 29000 nM T17345 CUOV62 135964392 IC50 > 34000 nM T17345 CG23QU 135964393 IC50 > 32000 nM T17345 CR5EG8 135964397 IC50 > 28000 nM T17345 C0T2QO 135964404 IC50 > 32000 nM T17345 CD8WY9 135964405 IC50 > 25000 nM T17345 CRXF18 135964411 IC50 > 31000 nM T17345 C87XGZ 135964413 IC50 > 32000 nM T17345 CF1N5G 136002190 IC50 = 750 nM T17345 C3LWJ1 136002235 IC50 = 460 nM T17345 CJ7ES6 136016316 IC50 = 290 nM T17345 C24FWM 136016317 IC50 = 370 nM T17345 C9SMI1 136016318 IC50 = 340 nM T17345 CMG1F8 136016319 IC50 = 300 nM T17345 C1GE3H 136016320 IC50 = 640 nM T17345 C56SPO 136046100 IC50 = 430 nM T17345 CT0NK9 136046104 IC50 > 40000 nM T17345 CA1R9P 136046152 IC50 = 950000 nM T17345 C6CMD5 136046154 IC50 = 1300 nM T17345 CDMI28 136056632 IC50 = 3800 nM T17345 CL8YP6 136056633 IC50 = 530 nM T17345 CZ0JY3 136056634 IC50 = 1500 nM T17345 CMQ87O 136056635 IC50 = 3800 nM T17345 C5X9UG 136078523 IC50 = 650 nM T17345 CTK4I6 136078526 IC50 = 260 nM T17345 CML42R 136092224 IC50 63300 nM T17345 C8O2GN 136109165 IC50 = 100 nM T17345 CALV20 136109177 IC50 = 100 nM T17345 CKI9N0 136136563 IC50 = 3000 nM T17345 CG3OA8 136136566 IC50 = 1400 nM T17345 C7QAB0 136171375 IC50 = 3200 nM T17345 C6XHI1 136171377 IC50 = 280 nM T17345 CVKL45 136171378 IC50 = 300 nM T17345 C23HGZ 136191424 Ki ~ 600 nM T17345 CVY71R 137300720 IC50 > 10000 nM T17345 CWE38X 137491959 IC50 = 12500 nM T17345 CM10NY 137631470 IC50 = 28000 nM T17345 CAZB89 137631503 IC50 = 2250 nM T17345 CWR72A 137632901 IC50 = 19000 nM T17345 CYF76S 137633375 IC50 = 5330 nM T17345 CFUY16 137633842 IC50 > 27000 nM T17345 CNT9K1 137634037 IC50 = 9.2 nM T17345 CZ5B9O 137634433 IC50 = 16900 nM T17345 CPB9Q3 137634556 IC50 = 1260 nM T17345 C0PNW5 137635062 IC50 = 450 nM T17345 CS23KQ 137635618 IC50 > 28000 nM T17345 CF5S9P 137636125 IC50 = 4 nM T17345 C7N6WS 137636390 IC50 > 150000 nM T17345 C53CKY 137636400 IC50 = 853 nM T17345 COE67T 137637328 IC50 > 50000 nM T17345 CL87FM 137638209 IC50 = 108 nM T17345 CA01DG 137638564 IC50 = 3.2 nM T17345 CP8X2O 137639098 IC50 = 290 nM T17345 CL95CK 137639545 IC50 = 6.1 nM T17345 CK6GP0 137640129 IC50 = 14800 nM T17345 C4QHY1 137640582 IC50 = 3610 nM T17345 C8MQ6U 137642178 IC50 = 2.6 nM T17345 C19WKB 137642364 IC50 = 6000 nM T17345 CU8YX6 137643005 IC50 > 27000 nM T17345 CW27XK 137644048 IC50 = 25000 nM T17345 C4N6GR 137644261 IC50 = 36 nM T17345 CT6CI1 137644294 IC50 = 710 nM T17345 C9YX2K 137644352 IC50 = 4000 nM T17345 CA7QW8 137645236 IC50 = 53.4 nM T17345 CSXF17 137645367 IC50 = 2840 nM T17345 CO0U6R 137646091 IC50 = 1400 nM T17345 C4NJB5 137646478 IC50 = 4.2 nM T17345 C83JEY 137646749 IC50 = 13.1 nM T17345 CRU6D2 137647615 IC50 = 5.3 nM T17345 CA7Y9F 137648264 IC50 = 4780 nM T17345 CZGU30 137648786 IC50 = 44 nM T17345 CQED79 137651284 IC50 = 2550 nM T17345 C5V4MO 137651590 IC50 = 14.1 nM T17345 CL1DZ0 137651595 IC50 = 5280 nM T17345 CQUY83 137652218 IC50 > 29000 nM T17345 CB3H5W 137652434 IC50 = 6.4 nM T17345 CSR07T 137654267 IC50 = 3190 nM T17345 CR71UO 137654559 IC50 = 950 nM T17345 C9JT1N 137655519 IC50 > 30000 nM T17345 C5XVK8 137656132 IC50 = 4130 nM T17345 C1M2YZ 137657601 IC50 = 2480 nM T17345 CQJD20 137657673 Ki = 13170 nM T17345 CX2T5K 137658038 IC50 = 35.6 nM T17345 CYV97X 137659199 IC50 = 4340 nM T17345 CO79SP 137659251 IC50 = 1670 nM T17345 CYML31 137659929 IC50 = 59.2 nM T17345 CETP42 137660220 IC50 = 3.4 nM T17345 C8W5GY 137660580 IC50 = 20100 nM T17345 C4UF6M 137660773 IC50 = 4.8 nM T17345 CD6VN2 137660870 IC50 = 9 nM T17345 C7V3LC 137661421 IC50 = 3.9 nM T17345 CFI5E0 137661591 IC50 = 18 nM T17345 CC8QH2 138460007 IC50 = 1090 nM T17345 C9NL0Q 138460276 IC50 = 1430 nM T17345 CL45VQ 145949793 Ki = 530 nM T17345 CX76CQ 145954183 Ki = 1400 nM T17345 C8QO7R 145955925 Ki = 640 nM T17345 CE0VX2 145967688 IC50 = 700 nM T17345 C49HWY 145967911 IC50 = 970 nM T17345 C4Q8MH 145968315 IC50 = 1101 nM T17345 CL72EN 145968368 IC50 = 1400 nM T17345 CK5H1X 145968380 IC50 = 579 nM T17345 C7ILN2 145968384 IC50 = 2730 nM T17345 CKC3W9 145968635 IC50 = 70510 nM T17345 C2V6SX 145968836 IC50 = 2318 nM T17345 CBP38L 145968849 IC50 = 590 nM T17345 C2LD6U 145968997 IC50 = 1917 nM T17345 CZ6LQ5 145969012 IC50 = 7930 nM T17345 C7N8WS 145969103 IC50 = 12290 nM T17345 CR9J7O 145970201 IC50 = 610 nM T17345 C04XEC 145970467 IC50 = 1130 nM T17345 C48KNM 145970614 IC50 = 811 nM T17345 CBXY67 145970730 IC50 = 2530 nM T17345 CT72GK 145970859 IC50 = 60 nM T17345 CIG4X8 145970868 IC50 = 11230 nM T17345 CHC2I0 145971065 IC50 = 2100 nM T17345 CEA95O 145971179 IC50 = 2046 nM T17345 CLY9F6 145988837 IC50 = 1104 nM T17345 CG36PF 145989276 IC50 > 100000 nM T17345 CUP4Z9 151456061 IC50 = 1360 nM T17345 CSL7O9 152598220 IC50 = 1790 nM T17345 C5OVQ3 152617142 IC50 = 347 nM T17345 CI79YB 155510882 IC50 = 1630 nM T17345 CB8J3L 155511255 IC50 = 37.94 nM T17345 C7GFM4 155512559 Ki = 18.41 nM T17345 CGK20J 155513582 IC50 = 819 nM T17345 C6D2CN 155514408 IC50 = 903 nM T17345 CS84IM 155515034 Ki = 555.55 nM T17345 CO9ZD7 155516975 IC50 = 29.29 nM T17345 CPX7N5 155517476 Ki = 23.42 nM T17345 CK8UH6 155518935 Ki = 13.41 nM T17345 C1ZA0M 155520729 IC50 = 1098 nM T17345 CHW46G 155523087 IC50 >= 1000 nM T17345 CUY38N 155523154 Ki = 18.24 nM T17345 CF4JM8 155523234 IC50 = 10 nM T17345 CEA02Z 155527030 Ki = 508.88 nM T17345 CT6S0G 155527248 IC50 = 237 nM T17345 CLO94T 155527394 Ki = 14.36 nM T17345 C3U4ED 155528338 IC50 = 300 nM T17345 C4N5QE 155528668 Ki = 19.55 nM T17345 C8PH3I 155529256 IC50 = 2626 nM T17345 C1GZ7W 155529285 Ki = 21.72 nM T17345 CR0O1S 155529844 IC50 > 30000 nM T17345 C87EWF 155530674 IC50 = 1100 nM T17345 CJ1P8L 155531623 IC50 = 1330 nM T17345 CT40PE 155532707 IC50 = 1800 nM T17345 C5H8LY 155532752 Ki = 32.89 nM T17345 C9OW3C 155533311 Ki = 74.16 nM T17345 C2P4MC 155534197 IC50 = 4125 nM T17345 C51XLA 155539843 Ki = 22.07 nM T17345 CFP3Y7 155540286 IC50 >= 1000 nM T17345 CG1S5K 155542983 IC50 = 65.88 nM T17345 C49SMW 155543062 IC50 = 2253 nM T17345 C0SNO1 155543141 IC50 = 3260 nM T17345 C5GZ1N 155543331 IC50 = 980000 nM T17345 CC20PV 155543847 IC50 = 1808 nM T17345 CP15AX 155544485 Ki = 48.67 nM T17345 C9MU3J 155546590 IC50 = 53.42 nM T17345 C9QN6E 155547319 IC50 = 100 nM T17345 CA4T8J 155548037 IC50 = 541 nM T17345 CNA65G 155549118 IC50 = 5980 nM T17345 CM5F3R 155550798 Ki = 8.72 nM T17345 CKBA16 155550915 IC50 = 973 nM T17345 C4SXE2 155551604 Ki = 32.43 nM T17345 CPV2I5 155552635 IC50 = 210 nM T17345 C2NIY4 155552687 Ki = 34.84 nM T17345 C3U7CK 155552787 IC50 = 1540 nM T17345 C0V2SW 155553051 IC50 = 125000 nM T17345 C1WXN8 155553663 IC50 = 2710 nM T17345 C4PLU8 155554619 Ki = 27.27 nM T17345 CVHM01 155555730 Ki = 12.5 nM T17345 C3KM4N 155556589 IC50 = 48.95 nM T17345 C4WH0C 155557612 Ki = 12.77 nM T17345 C8WB9O 155558582 IC50 >= 1000 nM T17345 CDB7F2 155560431 IC50 > 30000 nM T17345 CMYU10 155561126 Ki = 52.39 nM T17345 CE84AM 155561456 IC50 = 670 nM T17345 CXYW29 155562270 IC50 = 200 nM T17345 CU71YW 155562818 IC50 = 1571 nM T17345 CFM53Y 155563602 IC50 = 1576 nM T17345 CQ97VE 155565527 IC50 = 180000 nM T17345 C6COP9 155565754 IC50 = 1300 nM T17345 CV6WP8 155566484 IC50 = 9.28 nM T17345 C8BGX5 155567131 Ki = 29.05 nM T17345 CWON57 155567297 Ki = 45.97 nM T17345 C8M7LB 155567321 IC50 = 1338 nM T17345 CGMA98 155567948 Ki = 13.59 nM T17345 CUV9H3 155568251 IC50 = 2800 nM T17345 C9S2ON 155568330 IC50 = 468 nM T17345 C5ILH2 155568439 IC50 = 1373 nM T17345 D00IBG 643976 IC50 = 325000 nM T17345 D01HKU 44428667 IC50 = 120 nM T17345 D02ZCP 446244 IC50 = 620 nM T17345 D02ZPZ 6532431 Ki = 1.8 nM T17345 D03DRF 46886486 IC50 = 2000 nM T17345 D04PAW 16216218 IC50 = 250 nM T17345 D05WHM 6917908 IC50 = 4.4 nM T17345 D06DIH 158376 IC50 = 220 nM T17345 D06ERH 637760 IC50 > 100000 nM T17345 D06QEN 467889 Ki = 230 nM T17345 D06UPT 446752 IC50 = 4.3 nM T17345 D07LSP 135438608 IC50 = 1900 nM T17345 D07XLJ 462120 IC50 = 2400 nM T17345 D08GPU 490662 Ki = 2.9 nM T17345 D0B0UI 44428664 IC50 = 70 nM T17345 D0H8AW 291270 IC50 = 23000 nM T17345 D0J4KJ 446245 IC50 = 940 nM T17345 D0JY6J 93114 Ki = 10.4 nM T17345 D0LH5P 100516 IC50 = 4.1 nM T17345 D0ME8Z 24778025 IC50 = 0.39 nM T17345 D0O9YG 9049 Ki = 55.6 nM T17345 D0P9XE 46871716 Ki = 93 nM T17345 D0R4PS 135403648 Ki = 2370 nM T17345 D0S4ZT 46886512 IC50 = 5000 nM T17345 D0Y3TU 334409 Ki = 1 nM T17345 D0Z9QC 135517463 IC50 = 34 nM T17345 D0ZG7W 11441554 IC50 > 100000 nM T77393 C6F2WU 700755 Ki > 1000000 nM T77393 CZS6I0 720519 Ki > 1000000 nM T77393 CJL6Z8 765511 Ki = 323000 nM T77393 CQ2S4B 910123 Ki = 61000 nM T77393 C9AVC3 1006789 IC50 = 25000 nM T77393 C5XG0W 1006800 IC50 = 13620 nM T77393 C36IHN 1006808 IC50 = 24000 nM T77393 C3N7ZL 1006833 IC50 = 9630 nM T77393 CMD15J 1006856 IC50 = 22000 nM T77393 CA1X5I 1025961 IC50 = 22000 nM T77393 C3D1ZK 1266319 IC50 = 38000 nM T77393 CKR60Y 2810167 IC50 = 6000 nM T77393 CU0VC2 2943337 IC50 > 20000 nM T77393 CN9SE0 3308644 Ki = 843000 nM T77393 CAV9I1 3697667 Ki = 8440 nM T77393 C9FT3D 13430822 Ki = 589000 nM T77393 C9CR0M 15561337 Ki = 651000 nM T77393 C6C2JF 16483718 IC50 = 24000 nM T77393 C1XOL3 16487351 IC50 = 22000 nM T77393 CL3C9H 16645214 IC50 = 22000 nM T77393 C78LBG 16645215 IC50 = 30000 nM T77393 C4IAR3 16645216 IC50 = 12970 nM T77393 C6IM7Q 24757930 Ki = 27300 nM T77393 C6XPA0 39845054 IC50 = 48000 nM T77393 CC30IP 39845125 IC50 = 23000 nM T77393 CT4OS9 39845172 IC50 = 13000 nM T77393 CI9N1O 46864279 Ki = 120 nM T77393 CM51WO 46864280 Ki = 20 nM T77393 C81DFP 46866889 Ki = 200 nM T77393 C1U3KE 46867009 Ki = 3 nM T77393 CCKI47 46867010 Ki = 20 nM T77393 CT24XZ 46867121 Ki = 6300 nM T77393 C5WP7S 46867122 Ki = 7300 nM T77393 CM27BD 46867257 Ki < 1 nM T77393 CS6J9I 46889977 Ki = 160 nM T77393 C4DR8T 46889978 Ki = 30 nM T77393 CAJ5E1 46889979 Ki = 90 nM T77393 C8NY4I 46889980 Ki = 160 nM T77393 CK48PC 46889981 Ki = 80 nM T77393 CM5XP9 46889982 Ki = 27000 nM T77393 C0SFR4 46889983 Ki > 50000 nM T77393 C0L7GM 46889984 Ki = 3200 nM T77393 CPE06Y 46889985 Ki > 50000 nM T77393 CZ9VF6 46889986 Ki = 150 nM T77393 CXV0F2 46889987 Ki = 6500 nM T77393 COKG74 46889988 Ki = 1600 nM T77393 CP7E6H 46889989 Ki = 15100 nM T77393 CQTU62 46889993 Ki = 15000 nM T77393 CO7ZX4 46889994 Ki = 9000 nM T77393 C1WP0Q 46889995 Ki = 15600 nM T77393 C52WPZ 53356803 Ki < 1 nM T77393 C5JOC6 54766612 Ki < 1 nM T77393 CBT35C 54766613 Ki < 1 nM T77393 CH1KS7 70679466 IC50 = 338.2 nM T77393 C8IPK7 71586081 IC50 = 0.9 nM T77393 CY1J9L 85721372 IC50 > 20000 nM T77393 CN7F5K 127048565 IC50 = 660.9 nM T77393 C5J6QE 127048926 IC50 = 733.3 nM T77393 C9IK3M 127048927 IC50 = 127.4 nM T77393 CZ9T0Q 127048933 IC50 > 20000 nM T77393 C4DL6C 127048934 IC50 = 11400 nM T77393 CUN7F3 127048935 IC50 > 20000 nM T77393 CH1K3Y 127049251 IC50 = 206.1 nM T77393 CG84YX 127049252 IC50 = 207.2 nM T77393 CO0ZG4 127049253 IC50 = 130 nM T77393 C1IPG6 127049254 IC50 > 20000 nM T77393 CT10RI 127050095 IC50 > 20000 nM T77393 CL5V0S 127050385 IC50 = 1604 nM T77393 CXH7K0 127050386 IC50 = 198.5 nM T77393 C19BTR 127050387 IC50 = 465.7 nM T77393 C7T5WN 127052836 IC50 = 392.6 nM T77393 CC71PB 127052837 IC50 = 103.9 nM T77393 CBI1K8 127052955 IC50 > 20000 nM T77393 CO8X1P 127052956 IC50 > 20000 nM T77393 CR8JM3 127052957 IC50 > 20000 nM T77393 C75QVY 127052958 IC50 > 20000 nM T77393 CX8MA9 127052959 IC50 > 20000 nM T77393 CGY79B 127052960 IC50 > 20000 nM T77393 CQF37D 132580838 IC50 = 46.5 nM T77393 C0LHZ3 132580839 IC50 = 26.4 nM T77393 CN3MY7 134129874 IC50 > 20000 nM T77393 CVZS03 134129880 IC50 = 81.5 nM T77393 CO75BV 134129898 IC50 = 340.8 nM T77393 C15JEQ 134129903 IC50 = 13600 nM T77393 CSMF23 134129955 IC50 = 70.1 nM T77393 C8WNH1 134130001 IC50 > 20000 nM T77393 CZV10G 134130017 IC50 = 102.1 nM T77393 CMLA18 134130074 IC50 = 5800 nM T77393 C6OPH7 134130102 IC50 = 197.6 nM T77393 CZ9X1B 134130118 IC50 > 20000 nM T77393 CYO72F 134130195 IC50 = 47.9 nM T77393 C8M9NP 134130199 IC50 = 285.1 nM T77393 CN0HP5 134130274 IC50 = 104.6 nM T77393 C9DJC5 134130275 IC50 = 1363 nM T77393 C7A3FI 134130278 IC50 = 77.1 nM T77393 C1UR5D 134130359 IC50 > 20000 nM T77393 CL3Z2T 134130407 IC50 = 30.1 nM T77393 CO9BF6 134130408 IC50 = 1553 nM T77393 C9YS8H 134130465 IC50 = 92.5 nM T77393 CB08EV 134130500 IC50 = 62.5 nM T77393 CY24IA 134130560 IC50 = 113.4 nM T77393 C8XUN4 134130570 IC50 = 18.2 nM T77393 CRIW18 134130589 IC50 > 20000 nM T77393 CM5US2 134130592 IC50 = 8.5 nM T77393 CXH06K 134130734 IC50 = 285.3 nM T77393 CB61JP 134130757 IC50 = 7.6 nM T77393 C48BIF 134130903 IC50 > 20000 nM T77393 C5KRU7 134130925 IC50 = 75.8 nM T77393 CZ4J1P 134130945 IC50 = 95.6 nM T77393 CBP5O4 134130958 IC50 = 421.9 nM T77393 CYL7R9 134131003 IC50 = 88.7 nM T77393 CYFW16 134131026 IC50 = 50.2 nM T77393 CIN01V 134131045 IC50 = 15 nM T77393 CBF6E4 134131065 IC50 = 77.9 nM T77393 C4B7MN 134131117 IC50 = 3186 nM T77393 C59JMH 134131257 IC50 = 1093 nM T77393 CHJ39K 134131302 IC50 > 20000 nM T77393 C7GBH3 134131374 IC50 > 20000 nM T77393 C7SKU8 134131410 IC50 = 76 nM T77393 C3O4TN 134131411 IC50 > 20000 nM T77393 CF5S3O 134131548 IC50 = 70 nM T77393 C30GML 134131594 IC50 = 80.4 nM T77393 C56NTH 134135619 IC50 = 483.5 nM T77393 C17JRH 134135674 IC50 > 20 nM T77393 C7PN4W 134135702 IC50 = 263.5 nM T77393 C10RIC 134136312 IC50 = 1171 nM T77393 CCN03X 134137047 IC50 > 20 nM T77393 C3ZA5K 134137967 IC50 > 20 nM T77393 C71GIB 134140087 IC50 = 283.9 nM T77393 CB0NA6 134143014 IC50 = 162.4 nM T77393 C9IGQ2 134143930 IC50 > 20 nM T77393 C2RS6U 134144485 IC50 > 20 nM T77393 C3G6AQ 134145642 IC50 = 433.2 nM T77393 C9AJI4 134145666 IC50 > 20 nM T77393 C72APM 134148078 IC50 = 454 nM T77393 CO57LR 134148875 IC50 > 20 nM T77393 CG74JP 134149023 IC50 > 20 nM T77393 CCMR94 134149266 IC50 > 20 nM T77393 CRMX45 134149901 IC50 > 20 nM T77393 CG78KP 134153992 IC50 = 244.9 nM T77393 CF1KZ5 134155604 IC50 = 58.8 nM T77393 CI3CN5 134157644 IC50 = 811.6 nM T77393 CH1S6B 134364156 Ki = 3.53 nM T77393 C8LV1Q 134364178 Ki = 105 nM T77393 C4MIV7 134369551 Ki = 7540 nM T77393 CK6ZM1 134369552 Ki = 7210 nM T77393 C1OLR0 134369556 Ki = 665 nM T77393 CHNY14 134369557 Ki = 2600 nM T77393 C3LO6E 134369558 Ki = 17600 nM T77393 CLH26P 134369559 Ki = 219 nM T77393 C59CPA 134369560 Ki = 503 nM T77393 CJ3R0T 134369561 Ki = 3130 nM T77393 C12FZJ 134369563 Ki = 3910 nM T77393 C7QFN0 134369568 Ki = 690 nM T77393 CKUR59 134369576 Ki = 1380 nM T77393 C1Y3CD 134369579 Ki = 4130 nM T77393 C4F5BV 134369583 Ki = 1260 nM T77393 CK0JG5 134369594 Ki = 480 nM T77393 C0LKG2 134369619 Ki = 1460 nM T77393 CR6ZE1 134369620 Ki = 148 nM T77393 CYM14L 134369623 Ki = 118 nM T77393 C9Z7GJ 134369629 Ki = 42.5 nM T77393 CN8DO3 134369637 Ki = 27.6 nM T77393 CDVS67 134369647 Ki = 473 nM T77393 C3OE7I 134369648 Ki = 9.89 nM T77393 CLC39Q 134369650 Ki = 22.8 nM T77393 C71NAT 134369652 Ki = 28.9 nM T77393 CH8C7V 134369653 Ki = 76.1 nM T77393 C2C7AZ 134369665 Ki = 13.1 nM T77393 CT61JH 134369666 Ki = 185 nM T77393 CRW1A0 134369668 Ki = 184 nM T77393 CBW56J 134369669 Ki = 95 nM T77393 C6B9RO 134369670 Ki = 51.9 nM T77393 C4F1OP 134369672 Ki = 20.7 nM T77393 C15BUR 134369676 Ki = 2.82 nM T77393 CP46RA 134369681 Ki = 924 nM T77393 C63WBR 134369708 Ki = 16.4 nM T77393 C8B3LO 137349384 Ki = 85200 nM T77393 CSM61B 138319680 Ki = 0.044 nM T77393 CK27NV 138470399 Ki = 9.36 nM T77393 CMTD84 138470404 Ki = 65.1 nM T77393 CMG7V3 138470418 Ki = 2.51 nM T77393 CB24SI 138470423 Ki = 0.902 nM T77393 C8X5US 145981722 Ki = 109000 nM T77393 C9EAI7 145982119 Ki > 125000 nM T77393 CJ23AP 145988536 Ki = 1120 nM T77393 CF0BR7 145989019 Ki = 64000 nM T77393 C0IUB7 145989142 Ki = 117000 nM T77393 C49OYH 145990286 Ki > 125000 nM T77393 CK2C9E 145991249 Ki = 64300 nM T77393 C7YAG8 145992826 Ki = 118000 nM T77393 CX74VN 145992918 Ki = 29700 nM T77393 C2AHW4 145993387 Ki = 4.94 nM T49031 D00UVA 11556711 IC50 = 2.7 nM T49031 D01MML 49867936 IC50 = 8.44 nM T49031 D04AIT 5280445 IC50 = 1300 nM T49031 D0E7PQ 5311 IC50 > 25000 nM T49031 D0K8KX 5280343 IC50 = 2000 nM T49031 D0SH3I 387447 Ki = 0.55 nM T49031 D0T9TJ 3034010 IC50 > 100000 nM T49031 D05KED 53340666 IC50 > 25000 nM T49031 D07SDQ 969516 IC50 = 10000 nM T49031 D0DP0J 92135659 IC50 = 1670 nM T49031 D0F9BT 25067547 IC50 = 10 nM T49031 D0L4FS 5280961 IC50 = 9260 nM T49031 D0N0RN 11347535 IC50 = 22 nM T49031 D0U2BH 65064 IC50 = 86 nM T49031 D0VO0T 24800541 IC50 = 3 nM T49031 D0Y2SW 25183872 IC50 = 3 nM T49031 D0U7OU 3220 IC50 = 1220 nM T49031 CKGX24 7060 IC50 > 25000 nM T49031 C29BVT 11926 IC50 > 25000 nM T49031 CTK25Q 72277 IC50 = 1200000 nM T49031 CPSA65 80458 IC50 = 3000 nM T49031 CNIW58 107905 IC50 = 194 nM T49031 CDZ65K 199472 IC50 = 187 nM T49031 CA6ID2 241903 IC50 = 4580 nM T49031 C9A1KC 282849 IC50 > 25000 nM T49031 CF5T0S 282888 Ki = 2180 nM T49031 CPEL12 336327 IC50 > 100000 nM T49031 C46ZED 434315 Ki = 2120 nM T49031 C7HME8 439246 IC50 = 41600 nM T49031 C3YF4P 462382 IC50 = 1.2 nM T49031 C1MY6Z 490002 Ki = 2.3 nM T49031 CZ0AH3 638278 IC50 = 4880 nM T49031 C2DC6P 684753 Ki = 11500 nM T49031 CS4F8G 688857 IC50 = 5210 nM T49031 C2JU6P 833502 Ki = 10900 nM T49031 CS1P9Y 906456 IC50 = 172200 nM T49031 C2CR9F 1722365 Ki = 2010 nM T49031 C5FC0Z 2215326 IC50 = 3500 nM T49031 CL3KS0 5497183 IC50 = 61 nM T49031 CL9NX1 6610292 IC50 = 160 nM T49031 CK1U3G 6871286 IC50 > 10000 nM T49031 CL4VY9 9874885 Ki = 0.72 nM T49031 C3TDO0 9920246 IC50 = 1900 nM T49031 COK6X9 9960660 Ki < 1 nM T49031 CB2KX5 10032943 Ki = 0.5 nM T49031 CDPZ20 10099985 Ki = 5.7 nM T49031 C56PLQ 10258908 Ki = 0.72 nM T49031 CV25EX 10346881 IC50 = 51090 nM T49031 CO2HE7 10461001 Ki = 38 nM T49031 C5CBI2 10484581 Ki = 0.65 nM T49031 CDW5Y2 10542930 IC50 > 10000 nM T49031 CLU69K 10628969 IC50 = 420 nM T49031 CU8I1N 11243977 EC50 = 10 nM T49031 C1A2IM 11512726 IC50 = 2.9 nM T49031 C31TAR 11520347 Ki = 500 nM T49031 C6B5UF 11520360 IC50 = 52 nM T49031 C3GE9O 11532672 IC50 = 3360 nM T49031 CF2R5T 11534087 IC50 = 17 nM T49031 C61XQZ 11542118 IC50 = 1.5 nM T49031 CV56WA 11548000 IC50 = 6560 nM T49031 CWX6Y7 11549328 Ki = 32 nM T49031 C8MEH4 11549343 Ki = 140 nM T49031 C3BTN5 11556651 IC50 = 2.5 nM T49031 C2OPE1 11556685 IC50 = 2.4 nM T49031 CMH1V5 11563622 IC50 = 570 nM T49031 C8T5DM 11570453 IC50 = 170 nM T49031 C9KS5X 11578303 IC50 = 120 nM T49031 CB1L7I 11583999 IC50 = 260 nM T49031 CETS82 11585586 Ki = 45 nM T49031 CW7Z2P 11585713 IC50 = 2500 nM T49031 CH4RG7 11591941 IC50 > 10000 nM T49031 CFH34R 11598900 IC50 = 21000 nM T49031 CR9VG2 11599767 IC50 = 5.9 nM T49031 CKN7V8 11600122 Ki = 0.51 nM T49031 CO9PW8 11607192 IC50 = 78 nM T49031 CW0T9J 11613973 IC50 = 56000 nM T49031 C9OT1M 11621366 IC50 = 1.1 nM T49031 CX51NM 11636132 IC50 = 540 nM T49031 CB70KR 11636235 IC50 = 10 nM T49031 CLUA24 11636269 IC50 = 1400 nM T49031 CYR86V 11664755 IC50 = 49 nM T49031 CJFM60 11671614 IC50 = 4.3 nM T49031 CZ68VB 11672014 IC50 = 44 nM T49031 CZF9M1 11686028 Ki = 130 nM T49031 CE82UG 11692971 IC50 = 28000 nM T49031 CJE3N7 11693095 IC50 = 6.7 nM T49031 CJ1H4E 11700022 IC50 = 14 nM T49031 CX9D8R 11707332 IC50 = 2300 nM T49031 CF3Y2Q 11714595 IC50 = 49 nM T49031 CLBD57 15479395 IC50 = 220 nM T49031 C8D5OY 16084592 IC50 = 6670 nM T49031 C5RA8E 17480620 Ki = 7550 nM T49031 C7JCW4 21140132 Ki = 4700 nM T49031 C19EMT 23649126 IC50 = 700 nM T49031 CU0FE7 24752894 IC50 > 10000 nM T49031 C9E8MQ 24753965 IC50 = 7190 nM T49031 C7A4VT 24966905 IC50 > 10000 nM T49031 C5RCN7 24966906 Ki = 580 nM T49031 C1LJZ3 24966907 IC50 > 10000 nM T49031 C1MJ0W 25053219 IC50 = 1440 nM T49031 C64CJD 25111344 IC50 > 5000 nM T49031 CG52FR 42601513 Ki = 843 nM T49031 CB8H2Y 42612596 IC50 = 49 nM T49031 CN6D8U 44190246 IC50 = 4.37 nM T49031 CKH7Y0 44190247 IC50 = 1.6 nM T49031 CC8FG3 44191199 IC50 = 1.2 nM T49031 CKM83N 44307872 IC50 = 140 nM T49031 C21GXN 44410779 Ki > 450000 nM T49031 CXS71L 44411047 IC50 = 430 nM T49031 C90ZUI 44411546 IC50 = 2230 nM T49031 CMV46Q 44411707 IC50 = 4320 nM T49031 CP03SX 44411716 IC50 = 4150 nM T49031 CHFA42 44477958 IC50 = 15300 nM T49031 C69XJY 44477959 IC50 = 10000 nM T49031 C7NW5T 44555355 IC50 = 0.08 nM T49031 CN57MC 44583022 IC50 = 10 nM T49031 C9GUZ5 45140224 IC50 = 31 nM T49031 C5GAE4 45140225 IC50 = 3 nM T49031 C9RL7F 46233200 IC50 = 1 nM T49031 CNFQ84 46233201 IC50 = 2 nM T49031 CB57EF 46233202 IC50 = 100 nM T49031 CZ29GM 46233203 IC50 = 200 nM T49031 CQO52J 46233204 IC50 = 130 nM T49031 C4V9JP 46233205 IC50 = 300 nM T49031 C38TWK 46233206 IC50 = 524807460.3 nM T49031 CM81GQ 46864294 IC50 = 2.1 nM T49031 CX1YJ8 49799952 IC50 = 4.26 nM T49031 CHO3X2 49799953 IC50 = 7.63 nM T49031 C3XCL9 49859747 Ki = 2430 nM T49031 CIW0H6 50899478 IC50 = 0.55 nM T49031 C5QU2O 50899571 IC50 = 0.42 nM T49031 C8WD6E 50899573 IC50 = 0.39 nM T49031 CWDL81 52948098 IC50 = 16 nM T49031 C5EQD3 53362657 IC50 = 303.8 nM T49031 C7Q0RA 54455523 IC50 = 514 nM T49031 CV1P6X 56945245 IC50 = 92 nM T49031 CG2D5M 57149553 IC50 = 93 nM T49031 C3QG8L 59127842 IC50 = 1700 nM T49031 CLM1G5 60164712 IC50 > 30000 nM T49031 CGZ89B 65806958 IC50 = 24790 nM T49031 C82JTA 71305068 IC50 = 11600 nM T49031 CQD09I 71495550 Ki = 3744 nM T49031 CR38FB 71543331 Ki = 374.9 nM T49031 C2GAT5 71561597 IC50 = 1500 nM T49031 C62JWN 71561733 IC50 = 13000 nM T49031 CJ9AR2 71561735 IC50 = 5500 nM T49031 CXJP49 71561736 IC50 = 2800 nM T49031 CZ4I1N 71561866 IC50 = 10500 nM T49031 CHG65M 71561867 IC50 = 630 nM T49031 CA5T6O 71561868 IC50 = 2400 nM T49031 C2E9HV 71561869 IC50 = 480 nM T49031 C5FDT2 71561997 IC50 = 93 nM T49031 C2F0BJ 71561998 IC50 = 160 nM T49031 CSG26R 71561999 IC50 = 110 nM T49031 C45HOE 71562349 IC50 = 1200 nM T49031 CSDV65 71562351 IC50 = 1100 nM T49031 CKE98R 71625293 Ki = 101 nM T49031 CA95PY 71625294 Ki = 67 nM T49031 CVD0M7 71625412 Ki = 10.3 nM T49031 C6KP3Q 71625413 Ki = 10.8 nM T49031 CO9HD8 71625414 Ki = 11.4 nM T49031 CB7A3F 71625415 Ki = 10.6 nM T49031 CB24WG 71625416 Ki = 6 nM T49031 C6YL0H 71655218 IC50 = 38 nM T49031 CJ2B4Q 71655219 IC50 = 90 nM T49031 C58CEL 71655220 IC50 = 14 nM T49031 C4E2RB 71655221 IC50 = 5.7 nM T49031 C32PIH 71655289 IC50 = 35 nM T49031 C6BSW5 71655290 IC50 = 130 nM T49031 C19VOE 71655291 IC50 = 200 nM T49031 C6ZCI2 71655292 IC50 = 63 nM T49031 C7BIM2 71655353 IC50 = 29 nM T49031 CY78WU 71655354 IC50 = 230 nM T49031 C5H0IP 71655355 IC50 = 210 nM T49031 CW0Y5L 71655356 IC50 = 130 nM T49031 C8G6CQ 71655357 IC50 = 60 nM T49031 C2B4FJ 71655358 IC50 = 33 nM T49031 C1RYA4 71655419 IC50 = 300 nM T49031 C42YSR 71655420 IC50 = 57 nM T49031 CS3OP6 71655421 IC50 = 41 nM T49031 C7EW4B 71655422 IC50 = 47 nM T49031 C63MDL 71655423 IC50 = 30 nM T49031 CHCW60 71655482 IC50 = 28 nM T49031 C1Z7FJ 71655483 IC50 = 230 nM T49031 CZ0B7D 71655484 IC50 = 79 nM T49031 C75FOB 71655485 IC50 = 25 nM T49031 CQR98T 71655486 IC50 = 10 nM T49031 CM9U4L 71655547 IC50 = 77 nM T49031 CBMY45 71697266 Ki = 1620 nM T49031 CC1EV9 71697268 Ki = 260 nM T49031 CPW74Y 71697269 Ki = 800 nM T49031 CL0Q1G 71697270 Ki = 1450 nM T49031 CX1R7P 71697360 Ki = 300 nM T49031 C69BUX 71697361 Ki = 98 nM T49031 C2X5UT 71697363 Ki = 5900 nM T49031 C0UPY7 71697364 Ki = 440 nM T49031 C92HCM 71697365 Ki = 1340 nM T49031 CIPT74 71697366 Ki = 170 nM T49031 CJ52KP 71717087 Ki = 2.3 nM T49031 C7FLM2 72724741 IC50 = 50 nM T49031 CC65XM 72724804 IC50 = 28 nM T49031 C5IX8L 72724805 EC50 = 332 nM T49031 CK41SO 72724806 IC50 = 330 nM T49031 CR4A1Z 72724807 IC50 = 500 nM T49031 CJG3W2 73897219 IC50 = 63340 nM T49031 C0ER9W 74538726 IC50 = 5700 nM T49031 C1IN8Q 76310070 IC50 = 3380 nM T49031 CNYC80 76313773 IC50 = 1040 nM T49031 C0LU1D 76317291 IC50 = 900 nM T49031 C0U3XB 76317292 IC50 > 10000 nM T49031 CX6O8P 76317293 IC50 > 10000 nM T49031 CF8B7J 76320989 IC50 > 10000 nM T49031 CON57Y 76320990 IC50 > 10000 nM T49031 C3H2UI 76320991 Ki = 1100 nM T49031 CZO5L9 76320992 IC50 = 1660 nM T49031 C9P2HW 76320993 IC50 = 1650 nM T49031 CX5H3D 76320994 IC50 = 670 nM T49031 CP7R9O 76320995 IC50 = 1940 nM T49031 C1U5JY 76328224 IC50 = 1370 nM T49031 CN48JG 76328225 IC50 = 2190 nM T49031 CB89NY 76328226 IC50 = 800 nM T49031 CCF2T7 76328227 IC50 = 750 nM T49031 C4MAE1 76335476 IC50 = 580 nM T49031 CL30YE 76335477 IC50 = 2700 nM T49031 CG5E8R 76335478 IC50 > 10000 nM T49031 CV3S5J 76335479 IC50 = 1570 nM T49031 C4C2HT 76335480 IC50 = 1460 nM T49031 CQAL89 76335481 IC50 = 1660 nM T49031 CGY43C 78425867 IC50 = 2670 nM T49031 C0WA1V 86290925 Ki = 10260 nM T49031 C6FVI5 86302567 Ki = 560 nM T49031 C4T2MX 86302568 Ki = 330 nM T49031 CH1AU3 86302591 Ki = 1480 nM T49031 CNK78C 86302666 Ki = 0.14 nM T49031 CQLZ84 90381790 Ki = 39213 nM T49031 C0U9JN 90645047 Ki = 57 nM T49031 C9VK0E 90645048 Ki = 490 nM T49031 C8K2VQ 90645050 Ki = 85 nM T49031 CEN72L 90645051 Ki = 53 nM T49031 C4RAD1 90645052 Ki = 60 nM T49031 CJH69O 90645053 Ki = 4570 nM T49031 C54TGH 90645054 Ki = 80 nM T49031 C1EB8U 90645055 Ki = 2340 nM T49031 CFPT98 90655054 IC50 = 140 nM T49031 C5JZ8R 90655055 IC50 = 280 nM T49031 C3DWJ2 90655129 Ki = 8030 nM T49031 C5Z8EX 90655130 Ki = 10100 nM T49031 C6C2HX 90655131 Ki = 7670 nM T49031 C24PAH 90655132 Ki = 1450 nM T49031 CIXL21 90655133 Ki = 300 nM T49031 C2X7HV 90665951 IC50 > 1000 nM T49031 CRH4M3 90665952 IC50 > 1000 nM T49031 C5ZA4B 90665953 IC50 = 910 nM T49031 CPJ21F 90665954 IC50 = 50 nM T49031 C3KRH8 90665955 IC50 = 25 nM T49031 C1BA4E 90665956 IC50 = 12 nM T49031 CY80KV 90665957 IC50 = 8.4 nM T49031 CA48LV 90665958 IC50 = 5.4 nM T49031 CYB86O 90665959 IC50 = 22 nM T49031 CW8MS4 90665960 IC50 = 6.8 nM T49031 CQ67SO 90665961 IC50 = 4.8 nM T49031 CN94OJ 90665962 IC50 = 4.7 nM T49031 C2K9LZ 90665963 IC50 = 12 nM T49031 C81TAL 90665964 IC50 = 4 nM T49031 CP5S0X 90665965 IC50 = 3 nM T49031 C8IVK5 90665966 IC50 = 11 nM T49031 C7DL5F 90665967 IC50 = 3.7 nM T49031 C78ZBE 90665968 IC50 = 4 nM T49031 C2AG7C 90665969 IC50 = 3.9 nM T49031 C10CYW 90665970 IC50 = 1.1 nM T49031 CHBL08 90665971 IC50 = 940 nM T49031 CVZO36 90665972 IC50 = 22.6 nM T49031 C5EN3W 90665973 IC50 = 16 nM T49031 C62YEW 90665974 IC50 = 23 nM T49031 CF20ZD 90665975 IC50 = 160 nM T49031 CQE72G 90665976 IC50 = 7.3 nM T49031 CYF9H8 90665977 IC50 = 11.6 nM T49031 CJB32F 98103582 Ki = 17500 nM T49031 CG1IY3 98473743 Ki = 2350 nM T49031 C8NM0U 101553172 Ki = 2120 nM T49031 CG0N1O 101874275 IC50 = 16 nM T49031 CZX37E 102160215 IC50 = 14400 nM T49031 CVC0L7 102236951 IC50 = 93600 nM T49031 CXUQ14 102236952 IC50 = 31900 nM T49031 CHR18W 102579879 IC50 = 23600 nM T49031 C9C5OZ 117607839 IC50 = 782 nM T49031 C9BZ6E 117607841 IC50 = 185 nM T49031 CLHS74 117607901 IC50 = 926 nM T49031 CW9R0U 117607904 IC50 = 688 nM T49031 CKPU97 117607978 IC50 = 6630 nM T49031 C7QST8 117611788 IC50 = 6894 nM T49031 C2QDO6 117611839 IC50 = 54 nM T49031 CO1HJ9 117611880 IC50 = 18226 nM T49031 CZ6C1M 117611892 IC50 = 3620 nM T49031 C9YH1X 117611941 IC50 = 42468 nM T49031 C29AKS 118717990 IC50 = 0.38 nM T49031 CU4O3M 118718077 IC50 = 0.4 nM T49031 CS16DB 118718078 IC50 = 0.22 nM T49031 CK6E3L 118718085 IC50 = 0.34 nM T49031 CRZY67 118736272 IC50 = 290 nM T49031 CPY1S2 118736273 IC50 = 920 nM T49031 C2HWT3 118736382 IC50 = 17190 nM T49031 CY0VM1 118736383 IC50 = 12970 nM T49031 C6X0GY 118736384 IC50 = 13880 nM T49031 CS50HX 118736385 IC50 = 17310 nM T49031 C80ROJ 118736389 IC50 = 660 nM T49031 CIJ3E0 118736391 IC50 = 1630 nM T49031 CYO8P5 118736392 IC50 = 11730 nM T49031 C1DP4N 118899141 IC50 = 76000 nM T49031 CUH45I 118899149 IC50 = 78200 nM T49031 CA83ML 118899158 IC50 = 74870 nM T49031 C7YGZ8 122177663 IC50 = 360 nM T49031 CR80CE 122177664 IC50 = 930 nM T49031 CO0E6T 122189322 Ki = 3231 nM T49031 CG3U9I 122189323 Ki = 743.4 nM T49031 CM68CG 122189324 Ki = 7575 nM T49031 CWN52G 122189325 Ki = 906.2 nM T49031 CH08QC 122189326 Ki = 591.6 nM T49031 CSWG38 122189327 Ki = 951.9 nM T49031 C2ZJK1 122189328 Ki = 2113 nM T49031 CP7I6J 122189329 Ki = 963.1 nM T49031 CY7O0G 122189330 Ki = 1237 nM T49031 CO9E8A 122189331 Ki = 2347 nM T49031 CK7UV3 122189332 Ki = 1140 nM T49031 C8E7MQ 122189333 Ki = 1711 nM T49031 CI46QN 122189334 Ki = 949.8 nM T49031 CZ6LS4 122189335 Ki = 447 nM T49031 CZSI84 122189336 Ki = 385.2 nM T49031 C0OLW2 122204528 IC50 = 900 nM T49031 C90BKO 122520041 IC50 < 10 nM T49031 C3P0QD 122576697 IC50 = 220 nM T49031 C17FZG 127027248 IC50 = 26.24 nM T49031 C0DW3P 127027565 IC50 = 42.61 nM T49031 C6OVL9 127028490 IC50 = 49.5 nM T49031 CCF5E4 127028491 IC50 = 120.2 nM T49031 CV6JZ1 127028492 IC50 = 471 nM T49031 CO4D8I 127028814 IC50 = 24547089.16 nM T49031 C1Y9BP 127028815 IC50 = 3.34 nM T49031 CLB70K 127029400 IC50 = 8.32 nM T49031 C3FR6D 127029685 IC50 = 25.02 nM T49031 C6A1GD 127029686 IC50 = 4.6 nM T49031 CI6S1K 127030040 IC50 = 8.46 nM T49031 C4X7CO 127030041 IC50 = 2.34 nM T49031 C3LRH9 127030042 IC50 = 2.73 nM T49031 CAB69Z 127030043 IC50 = 16.4 nM T49031 CA50HP 127030044 IC50 = 114 nM T49031 C8DA4P 127030315 IC50 = 295120922.7 nM T49031 CQV32H 127030316 IC50 = 1.16 nM T49031 CI6P8J 127030317 IC50 = 1.15 nM T49031 CXQ69J 127030318 IC50 = 6.96 nM T49031 CQJ7F3 127030635 IC50 = 0.76 nM T49031 CZH53T 127030636 IC50 = 1.34 nM T49031 CO7WC6 127030637 IC50 = 2.46 nM T49031 CU0BJ3 127030638 IC50 = 862978547.8 nM T49031 C6Y2XQ 127031260 IC50 = 4.69 nM T49031 CJL9I1 127032443 IC50 = 1.02 nM T49031 CK3BX6 127032447 IC50 = 6.31 nM T49031 CI8RZ2 127032448 IC50 = 8.47 nM T49031 CV76UR 127032449 IC50 = 6.94 nM T49031 CVQ04L 127032450 IC50 = 4.82 nM T49031 CL36HN 127045979 IC50 = 26050 nM T49031 CI7H5T 127045980 IC50 = 23050 nM T49031 CIVH08 127045981 IC50 = 21540 nM T49031 C4ZG2O 127045982 IC50 = 16140 nM T49031 CWN9X5 127046160 IC50 = 14230 nM T49031 CUK8M7 127046161 IC50 = 13760 nM T49031 C4CAH2 127046162 IC50 = 13340 nM T49031 CDR54T 127047437 IC50 = 10250 nM T49031 CNL84P 127047438 IC50 = 17630 nM T49031 C3G7FU 127047439 IC50 = 9880 nM T49031 CED9T0 127047850 IC50 = 11860 nM T49031 C8QSW1 127048158 IC50 = 13800 nM T49031 CD51BP 127048159 IC50 > 25000 nM T49031 CP59LC 127048521 IC50 = 7800 nM T49031 CSLW65 127048522 IC50 > 25000 nM T49031 CADQ63 127048523 IC50 = 18700 nM T49031 C2A0UO 127048524 IC50 = 2300 nM T49031 CX65VA 127048525 IC50 = 21600 nM T49031 C5TS0O 127048526 IC50 > 25000 nM T49031 C3SY6Q 127049154 IC50 = 7600 nM T49031 CE5VT0 127049164 IC50 > 25000 nM T49031 CG9XP1 127049501 IC50 > 25000 nM T49031 CKYV35 127049817 IC50 > 25000 nM T49031 CVY2Q6 127049838 IC50 = 6300 nM T49031 CNX36Z 127049839 IC50 = 5600 nM T49031 COH67Z 127049840 IC50 = 9100 nM T49031 C1B4PE 127049841 IC50 = 5260 nM T49031 CJM29H 127049842 IC50 > 25000 nM T49031 CZIV95 127049843 IC50 = 15600 nM T49031 CDX7J4 127049844 IC50 = 5500 nM T49031 C3JE8G 127049845 IC50 = 6700 nM T49031 CEU1Y3 127050799 IC50 = 19200 nM T49031 CAS65J 127051646 IC50 = 8200 nM T49031 CLU6P9 127051647 IC50 > 25000 nM T49031 C9BFA0 127051648 IC50 > 25000 nM T49031 CMW2S6 127051649 IC50 > 25000 nM T49031 CE25WX 127051650 IC50 = 9900 nM T49031 C5REY7 127051651 IC50 > 25000 nM T49031 C4QXW2 127051652 IC50 > 25000 nM T49031 CL4N3G 127051653 IC50 = 8500 nM T49031 CFC43I 127052871 IC50 = 6100 nM T49031 C8AUE5 127053172 IC50 = 19900 nM T49031 C4YV1I 127053228 IC50 = 208929613.1 nM T49031 CPB1J8 127053229 IC50 = 3.21 nM T49031 CZR14W 127053267 IC50 = 4.18 nM T49031 CX53LM 127053268 IC50 = 1.12 nM T49031 CW3L9P 127053269 IC50 = 5.17 nM T49031 C6W2RO 127053272 IC50 = 524807460.3 nM T49031 C3AZ9G 127053273 IC50 = 5.24 nM T49031 CU8NW9 127053274 IC50 = 6.7 nM T49031 C4O6VG 127053280 IC50 = 162181009.7 nM T49031 C98AVC 127053285 IC50 = 1.26 nM T49031 CH2EP6 127053293 IC50 = 39 nM T49031 C3IVZ5 127053294 IC50 = 14.2 nM T49031 CDS47Y 127053295 IC50 = 17.2 nM T49031 CI2U8S 127053300 IC50 = 3.67 nM T49031 CQ6YW0 127053301 IC50 = 1.46 nM T49031 CT96PH 129047769 IC50 = 1140 nM T49031 CI24DQ 129047778 IC50 = 409 nM T49031 CI2J8F 129047830 IC50 = 110 nM T49031 C7BGS2 129047963 IC50 = 960 nM T49031 C4FRX1 132501288 IC50 = 26300 nM T49031 C34DQH 132501408 IC50 = 18500 nM T49031 CSP91A 132501468 IC50 = 5300 nM T49031 C1IFJ2 132501469 IC50 > 100000 nM T49031 CUT65O 132503175 IC50 = 370 nM T49031 CTQ8E6 132528967 IC50 = 2.4 nM T49031 CFB4V6 132528968 IC50 = 3 nM T49031 CM34ST 132528969 IC50 = 1.4 nM T49031 C5ZWQ8 132528970 IC50 = 4.3 nM T49031 C3WLQ2 134134387 IC50 = 15.7 nM T49031 CLM6F9 134134689 IC50 = 45.7 nM T49031 C5JS7V 134138393 IC50 = 669.9 nM T49031 CJ8ZN5 134139145 Ki = 420 nM T49031 C63QWU 134141164 IC50 = 16.9 nM T49031 C3EKC0 134142355 IC50 = 343.9 nM T49031 CEF0U1 134144291 IC50 = 601.4 nM T49031 CH9PI2 134146604 IC50 = 14.7 nM T49031 C8GH5D 134155148 IC50 = 152.9 nM T49031 C2Z5NM 134155499 Ki = 10980 nM T49031 C3K5UI 134155758 IC50 = 16.6 nM T49031 CH4XU1 134156052 IC50 = 23.7 nM T49031 C52IBY 134823859 IC50 = 394.2 nM T49031 C8VHK7 137632080 IC50 = 2710 nM T49031 CQO35X 137632519 IC50 = 2 nM T49031 CVSF43 137632662 IC50 = 25.7 nM T49031 C2NC9L 137633752 IC50 = 2180 nM T49031 CN78FJ 137633908 IC50 = 50 nM T49031 C08FKI 137634357 IC50 = 75 nM T49031 C3JI7B 137634520 IC50 = 5.5 nM T49031 CEJO70 137634807 IC50 = 510 nM T49031 CM3G2X 137635261 IC50 = 22160 nM T49031 CGPH59 137635270 IC50 > 1000 nM T49031 C40KOA 137635653 IC50 = 0.6 nM T49031 C64VSP 137636270 IC50 = 22290 nM T49031 C3H9XJ 137636488 IC50 = 41 nM T49031 CQP57Z 137636959 IC50 = 1 nM T49031 C3U2JC 137637883 IC50 > 50000 nM T49031 CW8D3F 137638026 IC50 = 197 nM T49031 C1HIY2 137638305 IC50 = 6.6 nM T49031 CNYU52 137639027 IC50 = 1.1 nM T49031 CZO8K2 137639142 IC50 = 5840 nM T49031 CNE56R 137639426 IC50 = 740 nM T49031 C0JQF2 137639470 IC50 = 39400 nM T49031 CG8V1S 137639601 IC50 = 3.8 nM T49031 CMK7O5 137639868 IC50 > 50000 nM T49031 CMSA73 137639962 IC50 = 260 nM T49031 C1KN9L 137640079 IC50 = 510 nM T49031 CVAK38 137640137 IC50 = 0.3 nM T49031 CB94IM 137640658 IC50 = 19600 nM T49031 CNVZ89 137640673 IC50 = 500 nM T49031 CIJ6E3 137640968 IC50 > 1000 nM T49031 C0B1FH 137641544 IC50 = 192.5 nM T49031 C6DF7U 137641807 IC50 > 1000 nM T49031 C0GWD7 137641958 IC50 = 10 nM T49031 CO1L4N 137642007 IC50 = 21.8 nM T49031 CH09CN 137642553 IC50 = 0.0002 nM T49031 C6DJF3 137642709 IC50 = 168 nM T49031 C3AEP5 137642951 IC50 = 99 nM T49031 CSXN16 137643018 IC50 = 44.25 nM T49031 CE0J4N 137643562 IC50 = 7 nM T49031 C0EY3T 137643629 IC50 = 2430 nM T49031 CB85DX 137643715 IC50 = 11.42 nM T49031 CJ6Z5F 137645427 IC50 > 1000 nM T49031 CL09KP 137645698 IC50 = 10 nM T49031 CEB8L5 137646135 IC50 > 50000 nM T49031 C5NF8R 137647268 IC50 = 90 nM T49031 CWOY74 137647871 IC50 = 1380 nM T49031 CC9R2E 137647922 IC50 = 2.6 nM T49031 C0KYZ2 137648206 IC50 = 237 nM T49031 CSF5N6 137648399 IC50 = 10.8 nM T49031 CNA75Z 137648431 IC50 = 8830 nM T49031 C7NYD8 137649498 IC50 > 1000 nM T49031 C19DEP 137649562 IC50 = 1360 nM T49031 C58EXC 137650165 IC50 = 200 nM T49031 CU9EK0 137650556 IC50 = 8.6 nM T49031 C7BUK5 137650655 IC50 = 12 nM T49031 CQ5AJ9 137650783 IC50 = 1.2 nM T49031 C7QW9D 137650914 IC50 = 57 nM T49031 C09QJA 137650983 IC50 = 1 nM T49031 C2NYK9 137651187 IC50 = 3 nM T49031 CCWZ51 137651207 IC50 = 20 nM T49031 CDQ41W 137651497 IC50 = 19.7 nM T49031 C04AZG 137651667 IC50 = 4 nM T49031 C57ZKC 137652515 IC50 = 182 nM T49031 C7R4DB 137653941 IC50 = 22 nM T49031 C8XLU1 137654027 IC50 = 29030 nM T49031 CGSU61 137654406 IC50 = 11.6 nM T49031 C2QMK8 137654413 IC50 = 40 nM T49031 CT08DG 137654519 IC50 = 1.5 nM T49031 CDAE50 137655349 IC50 = 23.17 nM T49031 CUC26W 137655738 IC50 = 20 nM T49031 CV8P6O 137656187 IC50 > 50000 nM T49031 CHV31Y 137656315 IC50 = 3570 nM T49031 CTA1F2 137656425 IC50 = 67 nM T49031 C90JMU 137656505 IC50 = 0.7 nM T49031 CSZ1A5 137657170 IC50 = 2.9 nM T49031 C1Y9RS 137657408 IC50 = 660 nM T49031 C5N2CB 137657727 IC50 > 1000 nM T49031 CNM6C4 137657944 IC50 > 1000 nM T49031 CJU5K7 137658335 IC50 = 110 nM T49031 CNFP69 137658811 IC50 = 2710 nM T49031 C3XE0H 137659182 IC50 = 0.9 nM T49031 CUFT31 137659572 IC50 = 17 nM T49031 CY6A3Q 137659779 IC50 = 18 nM T49031 C9CQ4N 137659903 IC50 = 25.93 nM T49031 CJQ6B7 137659959 IC50 = 3390 nM T49031 CY1S6E 137660489 IC50 = 24.58 nM T49031 C4BMO7 137660514 IC50 = 2 nM T49031 C8MH9V 137660779 IC50 = 18 nM T49031 CL1G7H 137661189 IC50 = 2.4 nM T49031 C01KBD 137661456 IC50 = 570 nM T49031 C1R9BC 137661627 IC50 = 13.3 nM T49031 CI96SM 137661745 IC50 = 1970 nM T49031 C1JH8K 138545006 IC50 > 100000 nM T49031 CLT78F 138545112 IC50 > 100000 nM T49031 C7DZ8K 138545235 IC50 > 100000 nM T49031 C5DJC6 138545265 IC50 = 10000 nM T49031 CIS28V 139209090 IC50 = 1412 nM T49031 CB46AI 139209092 IC50 > 100000 nM T49031 CMNL75 145960420 IC50 = 9.7 nM T49031 CL45BO 145960456 IC50 = 140000 nM T49031 C1W6TO 145960482 IC50 = 92 nM T49031 C0YF7Z 145960612 IC50 = 109 nM T49031 CU1EV5 145960693 IC50 = 126 nM T49031 C01WBE 145960929 IC50 = 335 nM T49031 C5G6LM 145961320 IC50 = 8900 nM T49031 C96AIF 145961391 IC50 > 100000 nM T49031 CI9QB0 145961558 IC50 = 210 nM T49031 CUIF27 145961566 IC50 = 10000 nM T49031 CQE07I 145961835 IC50 = 166 nM T49031 CI9JH6 145961877 IC50 = 6700 nM T49031 C3M4OD 145961898 IC50 = 18000 nM T49031 CBI7V1 145962019 IC50 = 27800 nM T49031 CN1I2C 145962168 IC50 = 69000 nM T49031 C8CSZ0 145962247 IC50 = 125000 nM T49031 CMD9X7 145962389 IC50 = 53 nM T49031 CVEF93 145962537 IC50 = 39000 nM T49031 C35NPT 145962676 IC50 = 192 nM T49031 C97URS 145962850 IC50 = 950 nM T49031 CVB9A4 145963178 IC50 = 36 nM T49031 CPA60M 145963188 IC50 = 65 nM T49031 CM95CN 145963260 IC50 = 155 nM T49031 CUL94O 145963403 IC50 = 275 nM T49031 COA19G 145963426 IC50 > 100000 nM T49031 C2LEB3 145963518 IC50 = 67000 nM T49031 CS6I8T 145964202 IC50 > 8000 nM T49031 CJ3Q5B 145964538 IC50 = 890 nM T49031 CKAS15 145964962 IC50 = 1100 nM T49031 CO83HL 145965095 IC50 > 8000 nM T49031 C15VCH 145966003 IC50 > 8000 nM T49031 C3L5IP 145966472 IC50 = 6300 nM T49031 C40QHP 145969617 IC50 > 8000 nM T49031 CV5NU9 145974241 IC50 = 2100 nM T49031 CQ42KP 145974420 IC50 > 8000 nM T49031 CRUD43 145974971 IC50 = 6100 nM T49031 CZ8H4Y 145975867 IC50 = 370 nM T49031 C38NRV 145976554 IC50 > 8000 nM T49031 CK2B4J 145978094 IC50 = 890 nM T49031 C9BWP4 145979302 IC50 = 2130 nM T49031 CN79HG 145979487 IC50 = 2800 nM T49031 CODE68 145979676 IC50 = 11.6 nM T49031 CEI3U1 145979850 IC50 = 4300 nM T49031 C24WEG 145980281 IC50 = 8.2 nM T49031 CIZU61 145980473 IC50 = 9.8 nM T49031 C35BOY 145980635 IC50 = 7.8 nM T49031 C69MQC 145980644 IC50 = 8.8 nM T49031 C07EJK 145980652 IC50 = 5.7 nM T49031 C5AYC4 145980811 IC50 = 64000 nM T49031 CG6UL0 145980995 IC50 = 1740 nM T49031 C2XPD3 145981337 IC50 = 2.7 nM T49031 C21VNK 145981642 IC50 = 22.8 nM T49031 CB67YT 145981691 IC50 = 1480 nM T49031 C41IRV 145981707 IC50 = 350 nM T49031 C5L8JM 145981943 IC50 = 12.9 nM T49031 CE94FB 145982013 IC50 = 7.7 nM T49031 C4UVP5 145982479 IC50 = 10.2 nM T49031 CLO3P1 145982669 IC50 = 74.86 nM T49031 C4B2NC 145982840 IC50 = 3.53 nM T49031 CL1F8N 145982922 IC50 = 28700 nM T49031 CGB54U 145983051 IC50 = 8.21 nM T49031 CQF0E2 145983505 IC50 = 4.16 nM T49031 CFE52X 145983530 IC50 = 27.75 nM T49031 C7SKN2 145983622 IC50 = 30.78 nM T49031 CG9LA8 145983719 IC50 = 5.89 nM T49031 C7WD8V 145983830 IC50 = 26.79 nM T49031 CSV4F0 145983965 IC50 = 20.44 nM T49031 C8WRQ7 145984091 IC50 = 21.17 nM T49031 C2UV4N 145984105 IC50 = 8.86 nM T49031 CPK4C5 145984357 IC50 = 4.82 nM T49031 C62OHN 145984529 IC50 = 5.26 nM T49031 CQ30LY 145984824 IC50 = 6.74 nM T49031 CF5R2L 145984944 IC50 = 3.22 nM T49031 CNZ16R 145985009 IC50 = 8.11 nM T49031 C16JLE 145985104 IC50 = 1.98 nM T49031 CVZ10A 145985697 IC50 = 42.79 nM T49031 C9G2VJ 145985757 IC50 = 387 nM T49031 C07VUG 145985780 IC50 = 2.31 nM T49031 C69VIS 145985988 IC50 = 593.7 nM T49031 CXBR78 145986043 IC50 = 12.89 nM T49031 C5X3GQ 145986425 IC50 = 6200 nM T49031 CRZE86 145986857 IC50 = 5100 nM T49031 CAJ5K8 145986961 IC50 = 3.6 nM T49031 CIB5Z9 145986993 IC50 = 5 nM T49031 CHWT73 145987085 IC50 = 6800 nM T49031 CM3H4F 145987197 IC50 = 2900 nM T49031 CNZ7R6 145987536 IC50 = 9200 nM T49031 CYBN31 145987734 IC50 = 835 nM T49031 C1EF3B 145988020 IC50 = 7.1 nM T49031 CM1U6F 145988104 IC50 = 15.9 nM T49031 CQIS01 145988427 IC50 = 6000 nM T49031 C4R3HC 145988596 IC50 = 7 nM T49031 CQ7W9S 145988601 IC50 = 13.2 nM T49031 CMW7U5 145989009 IC50 = 35.9 nM T49031 CN8K1E 145989337 IC50 = 3.1 nM T49031 CE16JH 145989568 IC50 = 113 nM T49031 CON2B3 145989641 IC50 = 7.7 nM T49031 CF3OZ9 145989730 IC50 = 18.7 nM T49031 CXG30R 145990249 IC50 = 11300 nM T49031 CWS03B 145991519 IC50 = 9.4 nM T49031 C8G1BT 145991875 IC50 = 10000 nM T49031 C8IL9E 145992200 IC50 = 5100 nM T49031 CBY18W 145992498 IC50 = 1400 nM T49031 CCU34H 145992780 IC50 = 360 nM T49031 C6GHQ9 145993211 IC50 = 22000 nM T49031 C2Q8BT 145993325 IC50 = 7.6 nM T49031 CVN3A5 145993374 IC50 = 6.6 nM T49031 CEVY70 145993649 IC50 = 880 nM T49031 CC24LD 145993770 IC50 = 19.7 nM T49031 CJO08K 145993925 IC50 = 125 nM T49031 C1UC2Z 147001460 IC50 = 77.1 nM T49031 CES1Y7 147009690 IC50 = 52.2 nM T49031 CYUM75 147335182 IC50 = 36.8 nM T49031 CSK1A5 147672609 IC50 = 4.6 nM T49031 CDX0I3 149045896 IC50 = 729 nM T49031 C1YFV0 155510465 IC50 < 10 nM T49031 CX74UV 155510547 IC50 < 10 nM T49031 C2AW9L 155510675 IC50 = 37 nM T49031 CLHB15 155510759 IC50 = 14 nM T49031 C4FH8S 155512766 IC50 = 48.3 nM T49031 C7J5BO 155512794 IC50 = 41.5 nM T49031 CZXI74 155513137 IC50 = 32 nM T49031 CL7I6A 155513548 IC50 = 30.8 nM T49031 C6IB7G 155513571 IC50 = 9 nM T49031 CY56QN 155514326 IC50 = 952 nM T49031 C5J0OF 155514653 IC50 = 253 nM T49031 C8E6ZX 155514792 IC50 = 1400 nM T49031 C0SDO2 155515259 IC50 = 230 nM T49031 CX76LO 155515463 IC50 = 34 nM T49031 CGW2M6 155516032 IC50 > 100000 nM T49031 C53ZEN 155516179 IC50 > 10000 nM T49031 CM3BV8 155516620 IC50 > 100000 nM T49031 CHU0Q9 155516696 IC50 = 111 nM T49031 C4VT1Y 155517101 IC50 = 430 nM T49031 C2BCH9 155517229 IC50 = 248 nM T49031 C6I7SU 155517529 IC50 = 154 nM T49031 CJ6ZU4 155517550 IC50 > 1000 nM T49031 CCB58J 155517652 IC50 = 481 nM T49031 CE95IQ 155518158 IC50 > 100000 nM T49031 CFQZ35 155518266 IC50 = 1410 nM T49031 CW8Z7I 155518578 IC50 = 8100 nM T49031 C5ATN1 155519023 IC50 = 232 nM T49031 C2OQU6 155519126 IC50 > 100000 nM T49031 CEF5D1 155519196 IC50 > 100000 nM T49031 C7FP0V 155519306 IC50 = 395 nM T49031 C5B4HU 155519323 IC50 = 14 nM T49031 CEJ56T 155519405 IC50 = 6700 nM T49031 CH9R4W 155520688 IC50 = 54 nM T49031 COL16B 155520712 IC50 = 8 nM T49031 C4WO3N 155521110 IC50 = 392 nM T49031 CNM0Q9 155521286 IC50 > 10000 nM T49031 CD4OH3 155521410 IC50 = 56 nM T49031 C0S4TP 155521499 IC50 = 30.6 nM T49031 CZKF54 155521690 IC50 = 1300 nM T49031 C8NOH2 155521815 IC50 = 6040 nM T49031 CJZT01 155522109 IC50 = 952 nM T49031 CTDK64 155522147 IC50 = 480 nM T49031 CN60CL 155522148 IC50 = 243 nM T49031 CB0WG8 155522381 IC50 = 2.1 nM T49031 C73DYM 155522560 IC50 = 5907 nM T49031 CQ3OD0 155522579 IC50 = 116 nM T49031 C8GNQ9 155522828 IC50 = 486 nM T49031 CM7ZA2 155523065 IC50 = 99 nM T49031 CW75YK 155523151 IC50 > 100000 nM T49031 CY3UP7 155523507 IC50 = 405 nM T49031 CL0IQ3 155523963 IC50 = 25.5 nM T49031 C94IEH 155524612 IC50 = 922 nM T49031 CZP1E6 155524975 IC50 = 30 nM T49031 CIP3E9 155526380 IC50 = 460 nM T49031 C5R3PX 155526504 Ki = 17 nM T49031 C78BVM 155526764 IC50 = 1130 nM T49031 CVJ70O 155526910 IC50 = 1561 nM T49031 CAC34Y 155527225 IC50 = 1800 nM T49031 COMG30 155527377 IC50 = 579 nM T49031 C6OC8R 155527614 IC50 = 836 nM T49031 CPHX68 155527880 IC50 = 1.5 nM T49031 CWZ17S 155528412 IC50 = 67 nM T49031 CROM71 155528428 IC50 = 436 nM T49031 C3PMD9 155529033 IC50 = 506 nM T49031 CW3G4Z 155529142 IC50 = 920 nM T49031 CCW71B 155529960 IC50 = 100 nM T49031 CYW5R1 155530452 IC50 > 100000 nM T49031 C2MW8Q 155530743 IC50 > 100000 nM T49031 CUP2B4 155531358 IC50 = 39 nM T49031 CIL2D0 155531506 IC50 = 51 nM T49031 CD84AS 155531896 IC50 = 40190 nM T49031 C9SH6Q 155532346 IC50 = 352 nM T49031 CLE8N1 155532865 IC50 = 660 nM T49031 CL9A0E 155532989 IC50 = 20.6 nM T49031 CK28QW 155533771 IC50 = 20 nM T49031 C2TR0X 155533978 IC50 = 50210 nM T49031 CEF08Q 155534115 IC50 > 100000 nM T49031 C9ODL6 155534328 IC50 = 968 nM T49031 CH9GO0 155534453 IC50 = 56.5 nM T49031 CG5E2L 155534840 IC50 = 16 nM T49031 C72EIY 155535051 IC50 = 89 nM T49031 C5G9LX 155535238 IC50 = 113 nM T49031 COZ5V6 155535430 IC50 = 46600 nM T49031 CT3A0N 155536062 IC50 = 14 nM T49031 C20BYW 155536148 Ki = 10.1 nM T49031 C9IL7E 155536781 IC50 = 38.8 nM T49031 C7O0SH 155537082 IC50 = 1111 nM T49031 CP7D4R 155537435 IC50 = 26.8 nM T49031 CCYI81 155537845 IC50 = 29370 nM T49031 C3EF7U 155538548 IC50 = 100 nM T49031 C2S5HL 155538665 IC50 = 52.1 nM T49031 C2NTI6 155538936 IC50 > 100000 nM T49031 CW5U4H 155539000 IC50 = 64.8 nM T49031 C6E1YP 155539344 IC50 > 100000 nM T49031 C69TOB 155539701 IC50 = 57 nM T49031 CLE9Y6 155539965 IC50 = 280 nM T49031 CT2V8E 155540850 IC50 = 4380 nM T49031 CTM03H 155540978 IC50 = 4726 nM T49031 C6RE8V 155540985 IC50 = 36.6 nM T49031 CQE43H 155541095 IC50 > 100000 nM T49031 C0T3CO 155541137 IC50 = 139.6 nM T49031 CNZ5B4 155541377 IC50 = 2000 nM T49031 C6OIY3 155541618 IC50 > 100000 nM T49031 C42XMS 155542291 IC50 = 3 nM T49031 C1K6NV 155542487 IC50 = 259 nM T49031 C41IBR 155542489 IC50 = 2200 nM T49031 CRU73P 155542979 Ki = 4.8 nM T49031 CHJY08 155543004 IC50 > 10000 nM T49031 CH92PY 155543085 IC50 = 1682 nM T49031 CH6X3Q 155543527 IC50 = 26 nM T49031 CTL46N 155543581 IC50 = 64 nM T49031 CB4K6P 155543584 IC50 = 274 nM T49031 C0EG5T 155543676 IC50 < 10 nM T49031 CR7WL1 155544072 IC50 = 35 nM T49031 C13HEG 155544089 IC50 > 10000 nM T49031 CH17XP 155544685 IC50 > 100000 nM T49031 C72ADE 155544797 IC50 = 162.2 nM T49031 CEC78A 155545362 IC50 > 1000 nM T49031 CB4J8F 155545830 IC50 = 162 nM T49031 C7YS2H 155546237 IC50 = 119 nM T49031 C3Q5GS 155546528 IC50 = 17 nM T49031 CV8T2E 155546596 IC50 = 269 nM T49031 C2R3FM 155546808 IC50 = 111.6 nM T49031 C0V4GT 155547050 IC50 = 2 nM T49031 CKY05M 155547055 IC50 = 37090 nM T49031 CBG9C3 155547430 IC50 = 98.2 nM T49031 CNS2J4 155548060 IC50 < 10 nM T49031 CQ0Z4K 155548281 IC50 = 35 nM T49031 C1LJ0G 155548285 IC50 = 257 nM T49031 CA8Z7D 155548324 IC50 = 9120 nM T49031 C8HVD1 155548349 IC50 > 100000 nM T49031 CZB82L 155548494 IC50 = 370 nM T49031 CC5H7R 155548878 IC50 > 100000 nM T49031 C8JC4L 155548940 IC50 = 50 nM T49031 CK4Q0J 155548955 IC50 = 3863 nM T49031 CX27NO 155549084 IC50 > 100000 nM T49031 CP7FQ0 155549178 IC50 > 1000 nM T49031 CIM5K2 155549227 IC50 = 39000 nM T49031 CH35KO 155550346 IC50 = 36 nM T49031 C12LPX 155551071 IC50 = 29 nM T49031 CRV20J 155551193 IC50 = 25 nM T49031 C6BZ4E 155551617 IC50 = 7 nM T49031 CCKN07 155551785 IC50 = 43.1 nM T49031 CX7P8L 155552184 IC50 = 853 nM T49031 CR7Q8D 155552542 IC50 = 2011 nM T49031 CH93MA 155553025 IC50 = 4.9 nM T49031 CBHM14 155553205 IC50 > 100000 nM T49031 C35NJC 155553210 IC50 = 45300 nM T49031 C2VBQ0 155553272 IC50 = 25 nM T49031 CK9FW3 155553273 IC50 = 60.7 nM T49031 CI15FC 155553565 IC50 = 8600 nM T49031 CVJ3E7 155553910 IC50 = 5000 nM T49031 C0DQC5 155554155 IC50 = 34.1 nM T49031 CDI56O 155554254 IC50 = 37.5 nM T49031 C1AIJ3 155554704 IC50 = 82070 nM T49031 C6YP0L 155554916 IC50 > 100000 nM T49031 C9GE3U 155554982 IC50 > 100000 nM T49031 C2IE7D 155555749 IC50 = 12430 nM T49031 CCI45A 155555926 IC50 = 361 nM T49031 C5SZB7 155556059 IC50 < 10 nM T49031 CJ0QX2 155556352 IC50 > 100000 nM T49031 CP58EH 155556856 IC50 = 26050 nM T49031 CW0K5V 155556875 IC50 < 10 nM T49031 CYJ92G 155557164 IC50 < 10 nM T49031 C6YSC7 155557266 IC50 < 10 nM T49031 C9M1NU 155557790 IC50 = 32 nM T49031 CXCF36 155558612 IC50 = 63 nM T49031 C0Z4ET 155558668 IC50 = 540 nM T49031 CK41QD 155558933 IC50 = 3.8 nM T49031 C5AQM2 155559051 IC50 < 10 nM T49031 CMH7V5 155559237 IC50 > 100000 nM T49031 CR3V7P 155559353 IC50 = 2.1 nM T49031 CT97AU 155559419 IC50 < 10 nM T49031 C7O2KR 155559420 IC50 = 638 nM T49031 CJ5UC9 155560661 IC50 = 33 nM T49031 C2GHS4 155561494 IC50 = 2.1 nM T49031 C98PWZ 155561783 IC50 = 1197 nM T49031 C5OM0U 155561976 IC50 = 12 nM T49031 CZJ52C 155562121 IC50 = 70450 nM T49031 CZXL78 155562443 IC50 = 530 nM T49031 CYB71Z 155563262 IC50 = 18 nM T49031 C2USA4 155563322 IC50 = 166 nM T49031 CZ3XY4 155563335 IC50 > 100000 nM T49031 C9CG3Y 155563835 IC50 = 189 nM T49031 C1UR9Y 155564187 IC50 = 118 nM T49031 CY83KQ 155564232 IC50 < 10 nM T49031 C3N8XZ 155564979 IC50 = 12030 nM T49031 C5YCE8 155565509 IC50 = 4 nM T49031 C0XSM3 155565602 IC50 = 44.9 nM T49031 CEAV80 155566012 IC50 = 5000 nM T49031 CV1L3T 155566407 IC50 > 10000 nM T49031 C7HP0L 155566550 IC50 = 770 nM T49031 CU53FD 155566562 IC50 = 49 nM T49031 CK87TX 155566958 IC50 = 21 nM T49031 C2T7GX 155567492 IC50 < 10 nM T49031 CT23WX 155567596 IC50 < 10 nM T49031 C5Z7YC 155567712 IC50 = 750 nM T49031 CG2KN0 155567727 IC50 > 100000 nM T49031 C7UPT8 155567911 IC50 = 127 nM T49031 CR1NB6 155568111 IC50 = 139 nM T49031 C63DVL 155568157 IC50 = 36.8 nM T49031 CIC1Q5 155568323 IC50 = 50.9 nM T49031 CV68GZ 155568757 IC50 = 1070 nM T49031 CUE8B1 155568787 IC50 = 205 nM T49031 C4ZV3Q 155568941 IC50 > 10000 nM T49031 C1I7QW 155568944 IC50 = 346 nM T49031 CL1QZ7 44583044 IC50 = 9 nM T49031 D00RIX 5280443 IC50 = 1800 nM T49031 D01NCW 11534772 IC50 = 460 nM T49031 D01UYI 5281607 IC50 = 4900 nM T49031 D05MDE 11505372 IC50 = 150000 nM T49031 D05VEV 11556056 IC50 = 120 nM T49031 D06NEB 11693148 IC50 = 35 nM T49031 D08AIJ 440735 IC50 = 14600 nM T49031 D09GZQ 11713852 IC50 = 1300 nM T49031 D09IMK 11621748 IC50 = 3.2 nM T49031 D0A5WN 11621347 IC50 = 2.1 nM T49031 D0B3US 11585523 IC50 = 3300 nM T49031 D0G3TK 5280863 IC50 = 10500 nM T49031 D0I0MU 11534625 IC50 = 69 nM T49031 D0K0KT 11621207 IC50 = 6.1 nM T49031 D0K4PY 114829 IC50 > 100000 nM T49031 D0M7BR 5280378 IC50 > 100000 nM T49031 D0Q4MO 23642227 IC50 = 150 nM T49031 D0QY3R 11513217 IC50 = 24 nM T49031 D0RB1V 6419835 IC50 = 124 nM T49031 D0RL4S 11714476 IC50 = 27 nM T49031 D0SY2M 5281708 IC50 > 100000 nM T49031 D0T3PW 5281672 IC50 = 10000 nM T49031 D0W3ON 416002 IC50 = 600 nM T49031 D0Y3TZ 370 IC50 = 7100000 nM T49031 D0Y6HD 90645049 Ki = 51 nM T00926 D0BP9C 193962 IC50 = 8500 nM T00926 D0K8KX 5280343 Ki = 2400 nM T00926 D0O3OS 104850 Ki = 1400 nM T00926 D0R0FE 2520 EC50 = 1925 nM T00926 D0R1RS 3715 IC50 = 12000 nM T00926 D0R3JB 4212 IC50 = 27.5 nM T00926 D0Z3DY 2333 Ki = 190 nM T00926 D02HTD 25167947 IC50 = 14900 nM T00926 D02QWY 24785538 IC50 = 36300 nM T00926 D0G7UX 5284373 EC50 = 1700 nM T00926 D0O2EF 56946615 IC50 > 100000 nM T00926 D0V7UQ 56946834 IC50 = 2500 nM T00926 D02VJY 3037617 IC50 = 5180 nM T00926 D07GTB 16760063 IC50 = 7570 nM T00926 C52MFS 1756 EC50 = 42000 nM T00926 C8C1JP 72343 IC50 = 38320 nM T00926 C5ZCH7 97332 IC50 = 26350 nM T00926 CL97OF 97548 IC50 = 9860 nM T00926 CA3NK8 193841 EC50 = 5100 nM T00926 CR67FB 243037 EC50 > 100000 nM T00926 CABJ72 276138 IC50 = 1760 nM T00926 CM70RQ 285815 IC50 = 16000 nM T00926 CN8ZL4 298546 EC50 = 45000 nM T00926 C7HME8 439246 Ki = 2400 nM T00926 COI2C9 560674 EC50 = 98000 nM T00926 CTF2J0 687260 EC50 > 100000 nM T00926 CH6MV7 715632 IC50 = 8770 nM T00926 C64RUF 877998 IC50 = 15900 nM T00926 CXR0P5 917533 IC50 = 8800 nM T00926 C7D1QN 921567 EC50 > 100000 nM T00926 CK8TP4 1019287 IC50 > 100000 nM T00926 CL27VW 1069464 IC50 = 3900 nM T00926 CXQ4P8 1183964 IC50 = 8130 nM T00926 CQT4J5 2094802 IC50 > 100000 nM T00926 C1A0FV 2298706 EC50 = 9800 nM T00926 CW6SA0 2787558 IC50 > 100000 nM T00926 C8PN0C 5280682 IC50 = 50000 nM T00926 CNI9X4 5281888 Ki = 600 nM T00926 CPHR19 5325373 EC50 > 100000 nM T00926 CJMT13 5325385 EC50 > 100000 nM T00926 C8VZ9T 5325386 EC50 > 100000 nM T00926 C81ZSW 5325387 EC50 = 85000 nM T00926 CTO51S 5352005 IC50 = 50000 nM T00926 CB2U6E 5467200 IC50 = 1100 nM T00926 C0EM5S 6509849 IC50 = 2800 nM T00926 C32UFI 9828452 IC50 = 61 nM T00926 C82UNW 9828532 IC50 = 1800 nM T00926 CI78PM 9848185 IC50 = 1050 nM T00926 C30DJS 9873998 IC50 = 800 nM T00926 CK5L6J 9904482 EC50 = 64000 nM T00926 CHI5S9 9975676 IC50 = 2900 nM T00926 CEG64W 9976758 EC50 = 2800 nM T00926 CDTB42 9979854 IC50 >= 250 nM T00926 CL5ZS9 9980860 IC50 = 650 nM T00926 C2B0CY 10004696 IC50 >= 250 nM T00926 CQI0Z7 10029563 IC50 = 76 nM T00926 C0HN4T 10031184 IC50 = 118 nM T00926 CG3RA9 10046544 IC50 = 1850 nM T00926 C5IQ2D 10047863 IC50 < 250 nM T00926 CK4A1L 10048669 IC50 = 1020 nM T00926 C2ZUK8 10051663 IC50 < 250 nM T00926 CC6U1G 10071405 IC50 >= 250 nM T00926 CSY05M 10072430 IC50 = 38 nM T00926 CO0QB1 10092403 IC50 = 7350 nM T00926 CWJ7R4 10094280 IC50 >= 250 nM T00926 CE6X4R 10221081 EC50 = 49100 nM T00926 C96LOC 10251349 IC50 > 50000 nM T00926 CQT7H4 10320818 IC50 = 65 nM T00926 C3I4DW 10322116 IC50 = 715 nM T00926 CY73KI 10322450 EC50 = 1800 nM T00926 CW6D4S 10333981 IC50 = 10800 nM T00926 CK9SQ7 10344755 IC50 = 533 nM T00926 CXG67L 10345205 IC50 = 500 nM T00926 C7Z4DU 10346312 IC50 >= 250 nM T00926 C7Z8IW 10379829 IC50 = 2870 nM T00926 CAO02N 10383921 IC50 = 789 nM T00926 CQU08N 10388318 IC50 >= 250 nM T00926 C36PIN 10407830 IC50 = 197 nM T00926 C1DYS4 10432300 IC50 = 920 nM T00926 CG40WP 10454772 IC50 = 910 nM T00926 CW4BK0 10455921 IC50 = 138 nM T00926 CE7IT1 10459316 IC50 >= 250 nM T00926 CCS90U 10472817 IC50 = 714 nM T00926 C78HZG 10495050 IC50 = 932 nM T00926 CE1U9A 10517005 EC50 > 100000 nM T00926 CCG5H3 10518339 IC50 = 14500 nM T00926 C8HWT1 10543161 IC50 = 2710 nM T00926 CD2EQ3 10585756 IC50 = 43100 nM T00926 CHE31J 10591449 IC50 > 100000 nM T00926 C58EFZ 10616146 IC50 = 4190 nM T00926 CH1V7U 10708375 IC50 = 20400 nM T00926 C7ANU6 10709061 IC50 = 8290 nM T00926 CH72SE 10709378 IC50 = 18300 nM T00926 CSK86O 10756523 IC50 = 2560 nM T00926 C01KTG 10758537 IC50 = 5970 nM T00926 CQF21J 10776189 IC50 = 26400 nM T00926 CI1RC8 10830017 IC50 = 4060 nM T00926 COHV95 10848828 IC50 = 4460 nM T00926 C53AIX 10850200 IC50 = 43400 nM T00926 C2BXZ1 11156535 IC50 >= 250 nM T00926 CKJ32I 11164648 IC50 = 6350 nM T00926 C5E8LY 11168500 IC50 = 20 nM T00926 C84PJK 11177283 IC50 = 94 nM T00926 C8HF7R 11177641 IC50 = 399 nM T00926 CYQ98P 11179994 IC50 = 138 nM T00926 CN3B9L 11186582 IC50 = 9000 nM T00926 CTBH70 11189272 IC50 = 2800 nM T00926 C8CWV4 11200621 IC50 = 632 nM T00926 C6XUE4 11201011 IC50 = 33 nM T00926 CLT87I 11212921 IC50 = 41 nM T00926 CFD6R7 11213871 IC50 = 48 nM T00926 CD8VO1 11214464 IC50 = 15 nM T00926 C63QRZ 11226516 IC50 = 17 nM T00926 C7PTZ8 11246811 IC50 >= 250 nM T00926 C79PBA 11247947 IC50 = 59 nM T00926 C86MWN 11249529 IC50 = 13.7 nM T00926 COJD26 11258566 IC50 = 2300 nM T00926 CEN76W 11261262 IC50 = 40.9 nM T00926 CI1M9O 11270541 IC50 = 28 nM T00926 CP13GR 11270563 IC50 = 59 nM T00926 C8NL3A 11281999 IC50 = 3440 nM T00926 C4I2ZV 11293873 IC50 = 2710 nM T00926 CY79US 11293906 IC50 = 110 nM T00926 CFX64S 11293909 IC50 = 166 nM T00926 CH7E1O 11293927 IC50 = 147 nM T00926 C1YH6T 11295806 IC50 = 97 nM T00926 CJYA49 11304370 IC50 = 24 nM T00926 CXKY42 11305058 IC50 = 45 nM T00926 CD9SN8 11316308 IC50 = 167 nM T00926 CE4HY2 11318194 IC50 = 88 nM T00926 CL8ZT6 11327691 IC50 = 3150 nM T00926 CY8G5H 11337594 IC50 >= 250 nM T00926 C78BGT 11339085 IC50 = 169 nM T00926 C65ZTX 11350733 IC50 = 820 nM T00926 C8P1QC 11351150 IC50 >= 250 nM T00926 CYZ51K 11359019 IC50 = 8370 nM T00926 C61ARN 11362459 IC50 = 1415 nM T00926 C31PLX 11376266 IC50 = 29 nM T00926 CZ9W0I 11385818 IC50 = 78 nM T00926 C8S3OV 11396606 IC50 = 87 nM T00926 C0G4AF 11408751 IC50 = 120 nM T00926 C13MRQ 11418752 IC50 = 955 nM T00926 CUO79V 11419244 IC50 = 63 nM T00926 C49LBJ 11432257 IC50 = 620 nM T00926 CTK09U 11443156 IC50 = 13 nM T00926 CLB97A 11443942 IC50 = 26.5 nM T00926 CM2J9W 11444700 IC50 < 250 nM T00926 CSK8F9 11453657 IC50 = 190 nM T00926 C19WQH 11454150 IC50 >= 250 nM T00926 CTQS76 11454703 IC50 = 10 nM T00926 C59DBU 11454819 IC50 < 250 nM T00926 CYCB17 11455462 IC50 = 107 nM T00926 C6W0MU 11477947 IC50 = 122 nM T00926 CH0T1B 11488138 IC50 = 27 nM T00926 CJXT34 11751643 IC50 = 67 nM T00926 CXWU95 11752839 IC50 < 250 nM T00926 C9X6DU 11774980 IC50 = 51 nM T00926 CLR59J 11775287 IC50 = 62 nM T00926 C2C3WI 11957988 IC50 > 20000 nM T00926 CG1CU7 12219475 EC50 > 100000 nM T00926 CS4D6C 12405466 EC50 = 15100 nM T00926 C4D7RX 12613559 EC50 = 26500 nM T00926 C6UJA5 13144102 EC50 > 100000 nM T00926 CT0DU8 13633111 IC50 = 20400 nM T00926 CO9ES2 13633119 IC50 = 1210 nM T00926 CJ9Z4M 15290116 EC50 = 72000 nM T00926 CLD92G 15999199 IC50 = 40600 nM T00926 C0A3IV 16092354 IC50 = 3730 nM T00926 CMVW98 16618023 EC50 = 728 nM T00926 CX06NR 17412108 IC50 = 39300 nM T00926 CB7T2K 20963109 IC50 = 7720 nM T00926 CFI13S 22310708 IC50 = 7820 nM T00926 CK4UG1 23323164 IC50 > 100000 nM T00926 C3ESV6 24178402 EC50 = 2800 nM T00926 C60EJI 25113688 EC50 = 9300 nM T00926 C6O2ZR 25225119 EC50 = 2700 nM T00926 C3J8PO 39176758 IC50 > 100000 nM T00926 CG7UZ6 44220872 IC50 = 12300 nM T00926 C8C9MJ 44220873 IC50 = 42600 nM T00926 CSLJ20 44220874 IC50 = 5380 nM T00926 CPIM70 44220875 IC50 = 21600 nM T00926 C01FMP 44220876 IC50 = 16200 nM T00926 C04ZKP 44220877 IC50 = 18300 nM T00926 CY9AW0 44221092 IC50 = 11600 nM T00926 C0X8OT 44221093 IC50 = 4510 nM T00926 C12MDG 44221095 IC50 = 14300 nM T00926 C3MNS1 44221096 IC50 = 27500 nM T00926 C2VWE1 44221097 IC50 = 1230 nM T00926 C9BNA1 44248179 EC50 = 73 nM T00926 CKA6N2 44276937 IC50 = 122 nM T00926 CTOA75 44368818 IC50 = 2020 nM T00926 CPLV23 44368900 IC50 > 10000 nM T00926 C26MFU 44368902 IC50 = 7600 nM T00926 CHO6P8 44368923 IC50 = 400 nM T00926 COWL28 44369026 IC50 = 1330 nM T00926 CDLX46 44369027 IC50 = 1560 nM T00926 C9VXD2 44369028 IC50 = 3840 nM T00926 CT0SK1 44369032 IC50 = 36000 nM T00926 CCD76W 44369044 IC50 = 37000 nM T00926 C1V6QO 44369052 IC50 = 900 nM T00926 CY08UQ 44369067 IC50 = 1000 nM T00926 C0FXA2 44369069 IC50 = 18570 nM T00926 C82JKC 44369082 IC50 = 1500 nM T00926 C0Z4TJ 44369087 IC50 = 15100 nM T00926 CZD46M 44369091 IC50 = 6350 nM T00926 CLIY42 44369110 IC50 = 1000 nM T00926 CTE65O 44369198 IC50 = 7200 nM T00926 C1J6DA 44369228 IC50 = 4500 nM T00926 CKPW47 44369229 IC50 = 3200 nM T00926 CA0PF4 44369232 IC50 > 100000 nM T00926 CU9H3K 44369247 IC50 = 39000 nM T00926 C05EUO 44369260 IC50 = 3330 nM T00926 CGU9Z8 44369264 IC50 = 2910 nM T00926 C5JLT0 44369265 IC50 = 2800 nM T00926 CE32OY 44369278 IC50 = 10000 nM T00926 C40XPZ 44404554 IC50 >= 250 nM T00926 CU97QG 44404555 IC50 < 250 nM T00926 CHX57V 44404558 IC50 < 250 nM T00926 C89BQU 44405535 EC50 = 420 nM T00926 CLV54W 44405572 EC50 = 250 nM T00926 C8A7CS 44405716 EC50 = 640 nM T00926 CM8O3W 44451264 EC50 > 100000 nM T00926 C45VCM 44451857 EC50 = 21000 nM T00926 CG61YX 44542293 EC50 > 100000 nM T00926 CI9VZ6 44542743 EC50 > 100000 nM T00926 C80EVI 44723582 EC50 > 100000 nM T00926 C43FNG 45266957 IC50 = 4180 nM T00926 C8C4ZS 45267881 IC50 = 22800 nM T00926 C8IYJ2 45268774 IC50 = 198000 nM T00926 CUE5Y2 45269621 IC50 = 29100 nM T00926 CJG13Y 45272176 IC50 = 24000 nM T00926 CAPW24 45272182 IC50 = 20700 nM T00926 COA30H 46227751 IC50 > 20000 nM T00926 CLWR13 46227752 IC50 > 20000 nM T00926 CX2EU1 46843551 EC50 = 13000 nM T00926 CON7Q5 46888534 EC50 = 46000 nM T00926 C53NLD 46888535 EC50 = 7610 nM T00926 CWO79T 46899560 EC50 = 12000 nM T00926 CUFI19 46899561 EC50 = 8700 nM T00926 C43WPR 46899562 EC50 = 8000 nM T00926 C2QX3P 46899563 EC50 = 63000 nM T00926 CBWT20 46899565 EC50 = 13600 nM T00926 CHR49C 46899724 EC50 > 100000 nM T00926 CZXN91 46899725 EC50 = 85800 nM T00926 C7ZS6E 46899726 EC50 = 29500 nM T00926 C1H9ML 56764960 IC50 = 22700 nM T00926 C2WYN9 56945196 IC50 > 100000 nM T00926 C7RW8P 56945197 IC50 = 11200 nM T00926 C7LDX6 56945198 IC50 > 100000 nM T00926 C2N8DS 56945199 IC50 > 100000 nM T00926 CN2WF6 56945201 IC50 > 100000 nM T00926 CB7W4E 56945202 IC50 > 100000 nM T00926 CT4BW6 56945299 IC50 > 100000 nM T00926 CTEJ21 56945300 IC50 = 45800 nM T00926 CU2HC7 56945301 IC50 = 40600 nM T00926 CUK5Q9 56945302 IC50 = 38800 nM T00926 C36HTV 56945303 IC50 = 46600 nM T00926 C7X2EU 56945304 IC50 = 44500 nM T00926 C4VNX9 56945305 IC50 = 16300 nM T00926 C1JCB9 56945418 IC50 = 44000 nM T00926 C6UD7F 56945419 IC50 = 32200 nM T00926 C98UJH 56945420 IC50 = 8000 nM T00926 C51PRX 56945421 IC50 = 22000 nM T00926 CES25H 56945422 IC50 = 9500 nM T00926 C2QB4L 56945423 IC50 = 7700 nM T00926 CA6UX7 56945524 IC50 = 74500 nM T00926 C4AVC1 56945525 IC50 = 40600 nM T00926 CC25LY 56945526 IC50 = 75800 nM T00926 C8KLW6 56945527 IC50 = 37900 nM T00926 C6ZSA3 56945528 IC50 = 30000 nM T00926 C2IAL8 56945529 IC50 = 28000 nM T00926 CP6G0O 56945530 IC50 > 100000 nM T00926 C27RQI 56946614 IC50 > 100000 nM T00926 CK1ZU5 56946616 IC50 = 23600 nM T00926 C73GCK 56946617 IC50 > 100000 nM T00926 CL8Z0F 56946723 IC50 = 23300 nM T00926 CIQ64Z 56946724 IC50 = 17200 nM T00926 CXMK07 56946726 IC50 > 100000 nM T00926 CRY4C6 56946727 IC50 = 80000 nM T00926 CV29FO 56946728 IC50 > 100000 nM T00926 CI69QT 56946831 IC50 > 100000 nM T00926 CDPU29 56946832 IC50 > 100000 nM T00926 C69ELZ 56946833 IC50 = 6100 nM T00926 CH7M4O 56946835 IC50 > 100000 nM T00926 CP1VK5 56951135 IC50 > 200000 nM T00926 C1XCE9 57393400 IC50 > 100000 nM T00926 CJXP74 71061793 EC50 > 100000 nM T00926 CA2N0L 71062020 EC50 = 31800 nM T00926 C0QGU2 71062093 EC50 = 33200 nM T00926 C5T0NL 71454923 IC50 = 11180 nM T00926 C4ZD2W 71492590 IC50 = 418 nM T00926 C0P6IG 71492759 IC50 = 434 nM T00926 CV9QS7 71524587 EC50 > 100000 nM T00926 C7JIG6 71524588 EC50 > 100000 nM T00926 C1EY6B 71524589 EC50 = 14700 nM T00926 C4LPZ3 71524590 EC50 = 3200 nM T00926 C60ZQJ 71524591 EC50 = 8800 nM T00926 CGV8F5 71525288 EC50 > 100000 nM T00926 CO9ZJ3 71560809 EC50 > 100000 nM T00926 C0E6OM 71560810 EC50 > 100000 nM T00926 C3T8ZF 71560811 EC50 > 100000 nM T00926 CFN89Y 71560812 EC50 > 100000 nM T00926 C42SMF 71560938 EC50 > 100000 nM T00926 C98LPJ 71560939 EC50 > 100000 nM T00926 CG8DU1 71618156 EC50 > 100000 nM T00926 C0Z3PN 71682039 EC50 > 100000 nM T00926 CV5Z9M 71682040 EC50 > 100000 nM T00926 C1IZT7 71682041 EC50 > 100000 nM T00926 COV12T 71682195 EC50 > 100000 nM T00926 C3Y4FW 71682196 EC50 > 100000 nM T00926 CLF3I8 71682197 EC50 > 100000 nM T00926 CN6Q3L 71696716 EC50 = 113 nM T00926 CQCF98 71724480 EC50 = 151 nM T00926 C1PR7Z 71724504 EC50 = 140 nM T00926 CA7K8Z 71724506 EC50 = 217 nM T00926 CD9KH7 71724532 EC50 = 250 nM T00926 CWR2L5 71724556 EC50 = 220 nM T00926 C4ODQ2 71724557 EC50 = 425 nM T00926 C7T0UM 71724558 EC50 > 1000 nM T00926 CUL9E2 71724582 EC50 = 238.3 nM T00926 CNW68B 71724606 EC50 = 616.7 nM T00926 CCZ9B3 71724628 EC50 = 230 nM T00926 C48CAR 72735227 IC50 = 14090 nM T00926 CQ5NB6 72950792 IC50 = 21800 nM T00926 CF57OZ 73346145 IC50 = 19000 nM T00926 CK3EX6 73355255 IC50 = 27500 nM T00926 C7NTB0 73356802 IC50 = 15100 nM T00926 CRB93S 89784681 EC50 = 301.7 nM T00926 CG71EX 89784708 EC50 = 175 nM T00926 C4ZOX6 89784717 EC50 = 670 nM T00926 C0ZQO6 89784722 EC50 = 171 nM T00926 C4U5CZ 89784733 EC50 = 208 nM T00926 CW17YB 89784735 EC50 = 272 nM T00926 C0VD4P 89784742 EC50 = 114 nM T00926 CZT7B9 89784751 EC50 = 135 nM T00926 CH70XJ 89784752 EC50 = 193 nM T00926 C6MRA2 89784753 EC50 = 87 nM T00926 C1JH4L 89784756 EC50 = 243.3 nM T00926 CN1RD8 89784760 EC50 = 333.3 nM T00926 C2YB6Q 89784818 EC50 = 137 nM T00926 CSK8X6 89784827 EC50 = 233.3 nM T00926 CENX80 89785043 EC50 = 103 nM T00926 CY46QV 89785047 EC50 = 172.3 nM T00926 CQL7T6 89785059 EC50 = 99 nM T00926 CENR59 89785064 EC50 = 263 nM T00926 CVZG56 89785117 EC50 = 78 nM T00926 CT43OU 89785127 EC50 = 133.8 nM T00926 C3FB6Q 89785132 EC50 = 219 nM T00926 C4S9WG 89785146 EC50 = 650 nM T00926 CCE95J 89785148 EC50 = 184 nM T00926 C9SBA1 89785178 EC50 = 246.7 nM T00926 CSI51G 89785190 EC50 = 225 nM T00926 CGB2P5 89785210 EC50 = 276.3 nM T00926 CTY1H5 89785238 EC50 = 155 nM T00926 CHGX10 89785254 EC50 = 292.7 nM T00926 CB1FR2 89794901 EC50 = 441.7 nM T00926 C43AXK 89795130 EC50 = 750 nM T00926 C70LJV 89795278 EC50 > 1000 nM T00926 CFU4W2 89795305 EC50 = 760 nM T00926 CVB23M 89795326 EC50 = 245 nM T00926 CX1W9Z 89795330 EC50 = 165 nM T00926 C7XG4U 89795333 EC50 = 950 nM T00926 C7W1TP 89795335 EC50 = 475 nM T00926 CAX9S0 89795337 EC50 = 457.5 nM T00926 COB3Z9 89795340 EC50 = 180 nM T00926 C6BW0Q 89795341 EC50 = 137.7 nM T00926 CUHC90 90469229 EC50 = 11900 nM T00926 C05JQB 90469230 EC50 = 7000 nM T00926 C41EMT 90469289 EC50 = 3900 nM T00926 CA1VH0 90469291 EC50 = 12400 nM T00926 C4NX2Q 90469293 EC50 = 6600 nM T00926 C0NW8T 90469355 EC50 = 5200 nM T00926 C8BRG2 101876951 EC50 = 1100 nM T00926 C0H9DF 101891699 EC50 = 23000 nM T00926 CXHQ89 102340685 IC50 = 4280 nM T00926 CJ7VI3 102340686 IC50 = 6260 nM T00926 CS1P5K 102340687 IC50 = 3380 nM T00926 C93SXK 102340688 IC50 > 100000 nM T00926 C86WSC 117777746 EC50 = 255 nM T00926 C9E0BT 117777811 EC50 = 135 nM T00926 C9YPJ7 117803128 EC50 = 579 nM T00926 C5GUV9 118708511 IC50 = 5800 nM T00926 CQLK93 118708512 IC50 > 100000 nM T00926 C5F8LY 118708513 IC50 = 13600 nM T00926 CL8H6M 118708514 IC50 > 100000 nM T00926 CCT4I2 118708515 IC50 > 100000 nM T00926 C7GI8W 118708516 IC50 > 100000 nM T00926 CE7Q3U 118708517 IC50 > 100000 nM T00926 C31MGA 118708518 IC50 > 100000 nM T00926 CKV6P1 118708519 IC50 > 100000 nM T00926 C1MJ4N 118708520 IC50 > 100000 nM T00926 C7WFJ3 118708521 IC50 = 2200 nM T00926 CVK89G 118708522 IC50 > 100000 nM T00926 C7G3ZV 118708523 IC50 = 94500 nM T00926 CG8S9M 118708524 IC50 = 15800 nM T00926 C9T4KE 118708525 IC50 = 11100 nM T00926 CG3LK4 118708526 IC50 = 8130 nM T00926 C42ETW 118708527 IC50 = 23600 nM T00926 C0OQ9P 118716252 EC50 = 41400 nM T00926 C3VRT8 118716258 EC50 = 5200 nM T00926 C4Z2DS 118719365 EC50 = 10000 nM T00926 CU6EP1 122179376 IC50 = 322 nM T00926 CIL20J 122179390 IC50 = 142 nM T00926 C0OUW1 122179391 IC50 = 141 nM T00926 CCE46L 126587406 EC50 > 1000 nM T00926 CZG92F 127028059 IC50 = 11300 nM T00926 CSR0Y7 127028060 IC50 > 100000 nM T00926 C8Z2XI 127028354 IC50 = 19800 nM T00926 C8Q9DG 127028355 IC50 = 20800 nM T00926 CRI72H 127028356 IC50 = 22700 nM T00926 C58QBI 127028357 IC50 > 100000 nM T00926 C6AIP3 127028358 IC50 > 100000 nM T00926 CG46ES 127028359 IC50 = 30100 nM T00926 CRP9U1 127028361 IC50 = 53300 nM T00926 CUC9I4 127040367 IC50 = 18500 nM T00926 C0I9VF 127040368 IC50 = 5500 nM T00926 CX9JE1 127040369 IC50 = 8300 nM T00926 CRM9W5 127040370 IC50 = 1800 nM T00926 CJY60W 127042304 IC50 = 58300 nM T00926 CO2P8K 127042305 IC50 = 26700 nM T00926 C56HDS 127042306 IC50 = 8300 nM T00926 CRI0X9 127042307 IC50 > 100000 nM T00926 CK4J8D 127042801 IC50 = 7300 nM T00926 C87PMI 127042802 IC50 = 13200 nM T00926 CRQ7U8 127042918 IC50 = 10900 nM T00926 CDL84X 127042919 IC50 > 100000 nM T00926 C39PWZ 127042920 IC50 = 38000 nM T00926 C21DSU 127042921 IC50 = 6800 nM T00926 C6UZ7C 127042922 IC50 > 100000 nM T00926 CSBM31 127042943 IC50 = 12100 nM T00926 C12BJD 127042944 IC50 = 18800 nM T00926 CZBJ54 127048170 IC50 = 1010 nM T00926 CO93BJ 127048171 IC50 = 8980 nM T00926 C6L0AF 127049502 IC50 = 636 nM T00926 CK1SN3 127049508 IC50 = 1070 nM T00926 CB9EV4 127049509 IC50 = 2500 nM T00926 C7PF5I 127050480 IC50 = 623 nM T00926 C59EXD 127050481 IC50 = 876 nM T00926 CUO40Y 127050796 IC50 = 910 nM T00926 C7MJ5X 127050797 IC50 = 586 nM T00926 CT6A2G 127050798 IC50 = 2360 nM T00926 C6V7JZ 127051981 IC50 = 418 nM T00926 C4P0LG 127051982 IC50 = 821 nM T00926 C5CX0B 127051983 IC50 = 200 nM T00926 CBQL62 127051984 IC50 = 340 nM T00926 C0FOG1 127051985 IC50 = 866 nM T00926 C1VP2D 127052887 IC50 = 9410 nM T00926 CG9TE5 127052888 IC50 = 643 nM T00926 CA7N9R 127052889 IC50 = 981 nM T00926 C6ZK3C 135449697 EC50 > 100000 nM T00926 CD2NR8 136110930 IC50 = 95000 nM T00926 C1EB8Q 136236384 EC50 > 100000 nM T00926 CI0KU2 137643961 IC50 = 15900 nM T00926 CHCB46 145956407 IC50 = 44200 nM T00926 C1F4LH 145971569 IC50 > 1000 nM T00926 CK61NI 145973976 IC50 > 1000 nM T00926 CF8L7A 145979103 EC50 = 298 nM T00926 C3EX7W 145979504 EC50 = 170 nM T00926 C4G7LT 145980033 EC50 = 95 nM T00926 C26OWY 145981942 EC50 = 156 nM T00926 C13VFZ 145985646 EC50 = 53 nM T00926 C4A1LN 145985882 EC50 = 38000 nM T00926 CI38SJ 145987174 EC50 = 28900 nM T00926 CFU24J 145987833 EC50 = 103 nM T00926 CGL02K 145988126 EC50 = 205 nM T00926 CX3YR7 145990226 EC50 = 200 nM T00926 CZRB08 145990960 EC50 = 62000 nM T00926 CN1V8K 145992500 EC50 = 208 nM T00926 CT02XU 145992768 EC50 = 121 nM T00926 CKZA78 145992770 IC50 = 12500 nM T00926 C07OTB 145993028 EC50 = 111 nM T00926 C65JUT 145993130 EC50 > 1000 nM T00926 C3UC5J 145994097 EC50 = 207.3 nM T00926 CKM79V 145994277 EC50 = 155.8 nM T00926 C5VRT4 155511477 IC50 > 100000 nM T00926 C1L0WJ 155511549 IC50 = 20000 nM T00926 CE4C1X 155512695 IC50 = 5800 nM T00926 C0AFT8 155514623 EC50 > 1000 nM T00926 CH6O3X 155515825 EC50 = 5080 nM T00926 CV9TF6 155516191 EC50 > 1000 nM T00926 C4IS7E 155518051 EC50 = 2200 nM T00926 CLQO05 155518383 IC50 = 9680 nM T00926 CA1BD2 155520579 EC50 = 12700 nM T00926 C8WFN9 155522227 IC50 > 100000 nM T00926 C8V3OE 155522345 IC50 > 100000 nM T00926 CQK86M 155522385 IC50 > 100000 nM T00926 CS18PU 155523410 EC50 = 5600 nM T00926 CN6ST7 155523417 EC50 > 1000 nM T00926 C86ZPR 155525910 EC50 = 4400 nM T00926 C8TQ4G 155526547 EC50 > 1000 nM T00926 C9BGT5 155528240 EC50 > 1000 nM T00926 C75OQS 155529248 IC50 = 2980 nM T00926 C3O4FR 155529325 IC50 > 100000 nM T00926 C56AHP 155530068 EC50 = 181.4 nM T00926 C9F3YI 155530680 IC50 = 44000 nM T00926 C6I0LU 155531567 IC50 = 18000 nM T00926 CUL2G4 155531672 EC50 > 1000 nM T00926 CJ5X8R 155532908 IC50 = 322 nM T00926 C4IW9M 155533366 EC50 = 5800 nM T00926 C9QT4A 155533532 IC50 = 85100 nM T00926 CHF7A6 155535686 EC50 > 1000 nM T00926 C28CPM 155536187 IC50 = 3600 nM T00926 CQC9E5 155536529 IC50 > 100000 nM T00926 CGM43D 155536878 IC50 = 40000 nM T00926 CYG84N 155537154 EC50 = 7300 nM T00926 C2J7TM 155537461 IC50 = 17300 nM T00926 CGD47O 155537584 EC50 > 1000 nM T00926 CNS83Y 155538210 IC50 = 33000 nM T00926 CVES34 155538494 EC50 = 1900 nM T00926 CLU37N 155539307 EC50 = 3000 nM T00926 CXN6C4 155539538 IC50 = 31000 nM T00926 CL6QG0 155542981 IC50 = 73000 nM T00926 C7JUC3 155543680 EC50 = 4500 nM T00926 C1HI5E 155550141 IC50 > 100000 nM T00926 CB8FC1 155550293 EC50 = 3500 nM T00926 C8B3LI 155551011 IC50 = 3700 nM T00926 CX43TI 155551742 IC50 = 41000 nM T00926 CIF4T8 155553306 EC50 > 1000 nM T00926 CEZ7B1 155554618 EC50 = 137 nM T00926 CX6CM0 155554919 EC50 = 530 nM T00926 CU9P0W 155555392 IC50 = 18000 nM T00926 C7JI4C 155555932 EC50 = 348.3 nM T00926 C27XQN 155558615 EC50 = 212 nM T00926 C8ATZ5 155558917 IC50 = 53000 nM T00926 CUNV65 155558919 EC50 > 1000 nM T00926 CFRS42 155559312 IC50 > 100000 nM T00926 CG6NC7 155560071 EC50 = 10100 nM T00926 CE6C4X 155562808 IC50 > 100000 nM T00926 CWM67C 155563340 EC50 = 2800 nM T00926 C6Z2XK 155566234 EC50 = 3700 nM T00926 CO1LU7 155567143 EC50 > 1000 nM T00926 C7KFG6 155567619 EC50 = 3900 nM T00926 CTV5K3 155568177 EC50 > 1000 nM T00926 C03SJY 155568508 EC50 = 139.3 nM T00926 CTXV81 155568869 EC50 > 1000 nM T00926 C0K1HQ 155569340 IC50 = 12900 nM T00926 D00RFY 5281612 IC50 = 3000 nM T00926 D00RIX 5280443 Ki = 2400 nM T00926 D01FGM 5280666 IC50 = 3000 nM T00926 D07NAY 5281692 Ki = 5000 nM T00926 D0G3TK 5280863 Ki = 2400 nM T00926 D0I7GE 11790 IC50 = 11300 nM T00926 D0T3PW 5281672 Ki = 2400 nM T17967 D03GFC 16741245 EC50 = 80 nM T17967 CHGI09 6597 IC50 = 9000000 nM T17967 CMC1D0 12892 Ki = 176 nM T17967 C6NQ9Y 1116656 IC50 = 3800 nM T17967 CHK89E 6102763 IC50 = 2000 nM T17967 C19DIZ 7178516 EC50 = 5200 nM T17967 CI5FC0 7178544 EC50 = 3800 nM T17967 CG7X9S 7178546 EC50 = 1100 nM T17967 CC28SV 16414363 IC50 = 10900 nM T17967 CHK6P1 16424570 IC50 = 5200 nM T17967 CKQY13 28361735 IC50 = 10500 nM T17967 C28NIL 29255080 IC50 = 1500 nM T17967 C80ODY 67932020 Ki = 1070 nM T17967 CXIN84 72376511 IC50 = 570 nM T17967 CELO13 72376512 EC50 = 456 nM T17967 C47XUW 86280454 IC50 = 65 nM T17967 CI7HO1 97281116 IC50 = 2500 nM T17967 CK6QG0 117972799 IC50 = 206 nM T17967 CUE2B5 118155888 IC50 = 1177 nM T17967 C2SA5C 118155890 IC50 = 416 nM T17967 C5CJ3D 118155894 IC50 = 154 nM T17967 C5Y8GW 118155895 IC50 = 432 nM T17967 C75WOG 118155906 IC50 = 195 nM T17967 C2OW7X 118155909 IC50 = 1196 nM T17967 C4QI2B 124201642 Ki = 2170 nM T17967 CRHZ85 124390110 IC50 = 7.8 nM T17967 C3FC0O 126200721 IC50 = 5900 nM T17967 C0VN5E 134561057 IC50 = 580 nM T17967 C46MPX 134561154 IC50 = 72 nM T17967 CKQ63N 134561155 IC50 = 58 nM T17967 C5X0YD 134561193 IC50 = 1514 nM T17967 CMQ04B 134561196 IC50 = 156 nM T17967 C30MTB 134561301 IC50 = 357 nM T17967 CHME32 134561302 IC50 = 67 nM T17967 C7WTU8 134561303 IC50 = 221 nM T17967 CR3V2E 134561305 IC50 = 65 nM T17967 CO3V2F 134561468 IC50 = 767 nM T17967 C8W3YG 136087021 IC50 = 1126 nM T17967 C0BUJ9 136249185 IC50 = 2600 nM T17967 CMO6K1 137636150 IC50 = 1657 nM T17967 CKU8P4 137638606 IC50 = 629 nM T17967 CAP1D8 137641886 IC50 = 1610 nM T17967 CS3KF0 137642154 Ki = 150 nM T17967 C7KIS8 137645507 IC50 = 1346 nM T17967 CSA49E 137646868 IC50 = 91 nM T17967 CI5TH3 137653481 Ki = 702 nM T17967 C7RB8J 137653507 Ki = 1330 nM T17967 C5XEM7 137655013 IC50 = 565 nM T17967 C0AZR8 137656816 IC50 = 68 nM T17967 C3SV7G 137659540 Ki = 1278 nM T17967 C9LP0W 137660248 IC50 = 4371 nM T17967 CHQ86U 149832647 IC50 = 140 nM T17967 CL6T4P 149986651 IC50 = 10 nM T17967 C24DWX 150179460 IC50 = 302 nM T17967 C7BM5V 150226583 IC50 = 126 nM T17967 CDO4W3 150362366 IC50 = 373 nM T17967 CJ17UR 150426809 IC50 = 18 nM T17967 CMS4L6 150703157 IC50 = 1620 nM T17967 C7J0AF 150821022 IC50 = 772 nM T17967 C1Z5DA 151004457 IC50 = 98 nM T17967 C02NBO 151026196 IC50 = 133 nM T17967 C0Q9PK 151406722 IC50 = 193 nM T17967 CY8OK4 151698036 IC50 = 110 nM T17967 C2RVC3 151777753 IC50 = 252 nM T17967 CKR2T1 151835909 IC50 = 113 nM T17967 CTI5R1 151961601 IC50 = 1455 nM T17967 CC3ME1 152131905 IC50 = 8 nM T17967 CAR6N3 152143591 IC50 = 132 nM T17967 C79SKI 152618834 IC50 = 184 nM T17967 C49BFR 155510663 IC50 = 2040 nM T17967 COH17B 155516961 IC50 > 10000 nM T17967 CRK41X 155523490 IC50 = 2660 nM T17967 C8K4NL 155527038 IC50 = 9910 nM T17967 CCG7K6 155528322 IC50 = 64 nM T17967 CNY40T 155534218 IC50 = 1960 nM T17967 CM20ZB 155534260 IC50 = 503 nM T17967 C8EH6M 155538895 IC50 = 95 nM T17967 C7BTJ9 155554053 IC50 = 8590 nM T17967 CA18GY 155563372 IC50 = 1660 nM T17967 C6Y5IM 155567964 IC50 = 7220 nM T89565 CV7IN2 104934 Ki = 210 nM T89565 C1KR5B 5327301 Ki = 98000 nM T89565 C37TKL 5327302 Ki = 12000 nM T89565 C64ZMN 5327304 Ki = 22000 nM T89565 C3IZ2W 5327307 Ki = 23000 nM T89565 C16DTL 5327308 Ki = 24000 nM T89565 C4O3QY 5327309 Ki = 63000 nM T89565 C3GUM7 5327310 Ki = 36000 nM T89565 CLAC59 9828058 Ki = 81 nM T89565 CDX7A4 10963183 Ki = 32000 nM T89565 CDT9G3 11467504 IC50 = 0.81 nM T89565 CJ57OA 14585243 Ki = 47 nM T89565 C8D5TB 44364680 Ki = 11000 nM T89565 C86ORE 44459987 IC50 = 13489.63 nM T89565 CDY2W5 49796910 IC50 = 0.2 nM T89565 CGY3W2 71471109 IC50 > 100000 nM T89565 CANH70 71716242 IC50 = 35200 nM T89565 C40WIR 71718085 IC50 = 750 nM T89565 CU75VK 71719897 IC50 = 19500 nM T89565 CBV6F1 71720507 IC50 = 560 nM T89565 CWM2E8 133081971 IC50 = 2980 nM T89565 CID3N6 134134572 Ki = 48 nM T89565 CV0R3B 134135432 Ki = 24 nM T89565 C3D7LQ 134136688 Ki = 59 nM T89565 CBY95D 134138690 Ki = 41 nM T89565 CG3EI1 134145896 Ki = 34 nM T89565 CI9X3K 134147411 Ki = 16 nM T89565 CP16IA 134148745 Ki = 111 nM T89565 CPE90G 134149983 Ki = 34 nM T89565 CBE39C 134151245 Ki = 135 nM T89565 CY0LD4 134152014 Ki = 59 nM T89565 C3K5HR 134153309 Ki = 28 nM T89565 CWQT79 134156687 Ki = 99 nM T89565 D0Y5IQ 44255320 IC50 = 5000 nM T50269 D00KHM 16362 EC50 = 1700 nM T50269 D01AZG 5073 EC50 = 320 nM T50269 D03YGR 156419 EC50 = 320 nM T50269 D09GDD 11167602 EC50 = 1800 nM T50269 D0A9YA 6918296 EC50 = 330 nM T50269 D0GQ7K 4046 EC50 = 2500 nM T50269 D0JC9N 60164 EC50 = 1300 nM T50269 D0K5WS 5280795 EC50 = 400 nM T50269 D0M8AB 750 EC50 = 94000 nM T50269 D0N6RF 65999 EC50 = 3200 nM T50269 D0P1FO 16078 EC50 = 1300 nM T50269 D0U5FS 3396 EC50 = 1200 nM T50269 D0Z5IU 1548887 EC50 = 380 nM T50269 D0Y2HR 2247 EC50 = 4200 nM T50269 C3O9AG 439709 EC50 = 12589.25 nM T50269 C8HZF2 783663 IC50 = 76 nM T50269 C9H1CE 5390854 EC50 = 590 nM T50269 C4SWU6 6324617 IC50 = 1700 nM T50269 C3W8ZK 17758335 IC50 > 100000 nM T50269 CH9J0Y 24846186 Ki = 67 nM T50269 COX8D7 44408895 IC50 > 100000 nM T50269 CR6CE1 44408940 IC50 > 100000 nM T50269 COY01R 44420834 IC50 = 3162.28 nM T50269 CE30WA 44420835 IC50 = 7400 nM T50269 C0DIM8 44420839 IC50 > 100000 nM T50269 CYE94N 44420840 IC50 > 100000 nM T50269 C59CNH 44420842 IC50 > 100000 nM T50269 C6N3DU 44420843 IC50 > 100000 nM T50269 C6Q1OE 44420847 IC50 > 100000 nM T50269 CKHC34 44420848 IC50 > 100000 nM T50269 C52YKX 44420851 IC50 > 100000 nM T50269 C23CLN 44420852 IC50 > 100000 nM T50269 C2NF6H 44420854 IC50 > 100000 nM T50269 CW2TL6 44420856 IC50 > 100000 nM T50269 C3XV2H 44420857 IC50 > 100000 nM T50269 CG30DJ 44420862 IC50 > 100000 nM T50269 C3AYZ8 44420865 IC50 > 100000 nM T50269 CVS4Z1 44420866 IC50 > 100000 nM T50269 CKG6M0 44420867 IC50 > 100000 nM T50269 CCB95G 44420868 IC50 > 100000 nM T50269 CYX7A3 44420870 IC50 > 100000 nM T50269 COH12C 44420871 IC50 > 100000 nM T50269 C9X7JH 44420872 IC50 > 100000 nM T50269 CR8HG1 44420875 IC50 > 100000 nM T50269 C19QZY 44420876 IC50 > 100000 nM T50269 CSZ5F4 44420878 IC50 = 2400 nM T50269 C6ZG0M 44420879 IC50 > 100000 nM T50269 C3IU8N 44420880 IC50 > 100000 nM T50269 CW80SJ 44420881 IC50 = 3981.07 nM T50269 CV8C2B 44420885 IC50 = 7943.28 nM T50269 CPBM16 44420891 IC50 = 3162.28 nM T50269 CYG93V 44427853 IC50 > 100000 nM T50269 C3C2OK 44427854 IC50 > 100000 nM T50269 C8Y9FW 44427856 IC50 > 100000 nM T50269 C19LSU 44427858 IC50 > 100000 nM T50269 C1FY4M 44427860 IC50 > 100000 nM T50269 CC2BE1 44427862 IC50 > 100000 nM T50269 CW95BM 44427864 IC50 > 100000 nM T50269 C3XJ4Z 44427866 IC50 > 100000 nM T50269 C84GXL 44427868 IC50 > 100000 nM T50269 C8CPX2 44427870 IC50 > 100000 nM T50269 CS17TJ 44427872 IC50 > 100000 nM T50269 CDL67C 44427876 IC50 > 100000 nM T50269 C9B6ER 44427877 IC50 > 100000 nM T50269 C15UHM 44427879 IC50 > 100000 nM T50269 CCAV10 44427881 IC50 > 100000 nM T50269 CXRV71 44427883 IC50 > 100000 nM T50269 CKX81C 44427885 IC50 > 100000 nM T50269 CG71DA 54467154 IC50 = 6900 nM T50269 C6DQT3 71450923 IC50 = 501.19 nM T50269 C2HUL4 90659973 IC50 > 100000 nM T50269 CO9ZU7 99118914 Ki = 40 nM T50269 CFW2V1 118195533 EC50 = 0.0012 nM T50269 CHM30C 118195560 EC50 = 0.06 nM T50269 C3HMN2 118195567 EC50 = 0.43 nM T50269 C8DSH5 118195581 EC50 = 0.00016 nM T50269 CKDM68 123133764 EC50 = 32 nM T50269 CPV2O3 132547348 EC50 = 327 nM T50269 CTN47D 135753560 IC50 = 8800 nM T50269 C8H3QG 135753564 IC50 > 200000 nM T50269 CLE71N 137631631 IC50 = 109 nM T50269 CL2X3J 137631882 IC50 = 690 nM T50269 C4L8SF 137635401 IC50 = 260 nM T50269 C1YE3F 137637510 IC50 = 720 nM T50269 CS41FM 137639832 IC50 = 4590 nM T50269 CKR79P 137644791 IC50 = 165.96 nM T50269 CVL25O 137645081 IC50 = 245.47 nM T50269 C3DZ4I 137650620 IC50 = 49 nM T50269 CDP0F7 137654599 IC50 = 220 nM T50269 C5QN0I 137655067 IC50 = 380.19 nM T50269 CU8FI4 137656578 IC50 = 75 nM T50269 CF1C3T 137657339 IC50 = 51.29 nM T50269 CRZY05 155519552 Ki = 741 nM T50269 CF27SE 155541454 Ki = 91 nM T50269 D04IEW 9909368 IC50 = 1900 nM T50269 D0H0BD 441071 Ki = 23 nM T50269 D0M4ZK 44420890 IC50 = 5011.87 nM T50269 D0X3TL 44420886 IC50 = 6200 nM T67710 D02CII 76943386 EC50 = 0.02 nM T67710 D03NHS 76283707 EC50 = 4100 nM T67710 CA6P1K 11963968 Ki = 0.912 nM T67710 CA4WI0 12001598 Ki = 707.95 nM T67710 CNF70V 16220269 IC50 = 68000 nM T67710 CH3KU5 23626097 Ki = 2818.38 nM T67710 CF1V4U 23626240 Ki = 3388.44 nM T67710 C5K7RJ 23626241 Ki = 562.34 nM T67710 C7O1ZX 23626243 Ki = 676.08 nM T67710 CS2FX3 23626399 Ki = 288.4 nM T67710 C0ZIC4 23626400 Ki = 154.88 nM T67710 CSI39A 23626402 Ki = 70.79 nM T67710 C0XE1Q 23626403 Ki = 3.802 nM T67710 CUTB14 23626557 Ki = 13.18 nM T67710 C5TJF3 23626558 Ki = 50.12 nM T67710 C0LNV5 23626559 Ki = 20.42 nM T67710 C27CIX 23626560 Ki = 6.761 nM T67710 CXU8E9 23626561 Ki = 3.548 nM T67710 C7JG9E 23626730 Ki = 1.445 nM T67710 C5N9AK 23626731 Ki = 1.82 nM T67710 CF8X4T 23626732 Ki = 6.761 nM T67710 C3B8PO 23626733 Ki = 616.6 nM T67710 CF4NW8 23626734 Ki = 8.71 nM T67710 CVO15W 23626891 Ki = 6.607 nM T67710 CB3D4J 23626894 Ki = 83.18 nM T67710 CU75YI 25118026 IC50 = 9400 nM T67710 CC9G1A 44270419 EC50 = 7.9 nM T67710 CS9AC3 44270511 EC50 = 4.4 nM T67710 C02OVQ 44270512 EC50 = 5.5 nM T67710 CC1OX8 44270513 EC50 = 9.1 nM T67710 CN3D6A 44428088 Ki < 100000 nM T67710 CPY82C 44428090 Ki = 933.25 nM T67710 CRS3H8 44428091 Ki = 380.19 nM T67710 C4FXJ3 44428092 Ki = 112.2 nM T67710 CN6WS7 44584917 EC50 = 32 nM T67710 CH14QN 44584920 EC50 = 13 nM T67710 CJR45V 44584921 EC50 = 0.06 nM T67710 CXSB17 44584922 EC50 = 0.15 nM T67710 CQS1U6 45485585 EC50 > 10000 nM T67710 C5XME6 49838154 EC50 > 1000000 nM T67710 C09VXY 49840922 EC50 = 1122 nM T67710 CPX2V6 49841000 EC50 = 0.2 nM T67710 CU3J0E 50908590 EC50 = 2.4 nM T67710 C24IPZ 56841901 EC50 = 0.07 nM T67710 C6Y8QI 66815925 EC50 > 1000000 nM T67710 CM8BP9 66817107 EC50 = 26000 nM T67710 C6IP4J 66817215 EC50 = 32000 nM T67710 CVCF27 66817553 EC50 = 33000 nM T67710 CAX82O 66817788 EC50 = 12000 nM T67710 C6CM8L 76283959 EC50 = 3600 nM T67710 C4WM1Z 137631923 EC50 = 19 nM T67710 C9XVZ4 137634846 EC50 = 0.51 nM T67710 CHV35B 137634885 EC50 = 0.26 nM T67710 CWA3V8 137635204 EC50 = 1.12 nM T67710 CIN0J6 137635394 EC50 = 0.08 nM T67710 CB64NJ 137636149 EC50 = 0.15 nM T67710 CP59IE 137636311 EC50 = 0.51 nM T67710 C7KQ9X 137637857 EC50 = 0.29 nM T67710 C6ZXO0 137637950 EC50 = 3 nM T67710 CLW1R3 137639371 EC50 = 14.57 nM T67710 CUZP78 137639372 EC50 = 0.13 nM T67710 C7O9IM 137639587 EC50 = 18.69 nM T67710 C05BRV 137640122 EC50 = 0.52 nM T67710 CT9B3U 137640833 EC50 = 0.34 nM T67710 C1O3FE 137641949 EC50 = 0.4 nM T67710 CSY1M3 137642287 EC50 = 0.14 nM T67710 C93LST 137642401 EC50 = 4.98 nM T67710 C3V6MW 137642849 EC50 = 0.12 nM T67710 C12BTY 137643019 EC50 = 0.34 nM T67710 CDR83Q 137643296 EC50 = 1.8 nM T67710 CQIU59 137645140 EC50 = 0.71 nM T67710 C71AOQ 137650056 EC50 = 11.51 nM T67710 C89VPB 137651582 EC50 = 0.18 nM T67710 C4A9EI 137652688 EC50 = 9.74 nM T67710 CL41NK 137654722 EC50 = 0.36 nM T67710 CV6G8Y 137657562 EC50 = 1.84 nM T67710 CRNM53 137657563 EC50 = 167 nM T67710 C79QHV 137657564 EC50 = 0.44 nM T67710 CN6V0J 137657565 EC50 = 0.83 nM T67710 CE0J2B 137657566 EC50 = 0.79 nM T67710 CQ8J3B 137657687 EC50 = 0.32 nM T67710 C5Q7KC 137657688 EC50 = 0.65 nM T67710 C38QDU 137657689 EC50 = 4.13 nM T67710 C5PM6C 137659455 EC50 = 0.48 nM T67710 CE5MN9 137659482 EC50 = 0.06 nM T67710 C3BK4S 137659489 EC50 = 2.59 nM T67710 C0ZJN1 137659716 EC50 = 0.17 nM T67710 C4TH5F 137660321 EC50 = 9.84 nM T67710 C8WFK3 137660410 EC50 = 0.27 nM T67710 CCT8K0 139035050 IC50 = 90 nM T67710 CDXQ89 145964425 EC50 = 67000 nM T67710 C60ZAH 145975286 EC50 = 50000 nM T67710 C9MJG6 145975813 EC50 > 1000000 nM T67710 CL3X2U 155513348 EC50 = 4600 nM T67710 C26GUZ 155518374 IC50 = 6800 nM T67710 CXZ5W0 155521869 IC50 > 100000 nM T67710 CB7Z3X 155522420 IC50 = 3500 nM T67710 CX2TS6 155522839 IC50 = 7600 nM T67710 CN5D9T 155526572 IC50 = 6100 nM T67710 C8LAP0 155529306 IC50 > 100000 nM T67710 CAE4T8 155533095 EC50 = 3600 nM T67710 CKW9P0 155536792 EC50 = 2.5 nM T67710 CTQ9U5 155536860 IC50 = 14000 nM T67710 C2I0PA 155540108 IC50 = 14000 nM T67710 CHM51V 155542161 EC50 = 5300 nM T67710 C2BHW9 155543526 IC50 = 38000 nM T67710 CGT23X 155546261 IC50 = 730 nM T67710 C59QIA 155547998 IC50 = 2300 nM T67710 C38KWY 155550447 IC50 = 4100 nM T67710 CGS61H 155551285 IC50 = 44000 nM T67710 CQ7ZP6 155553639 EC50 = 4600 nM T67710 C65GPR 155553648 EC50 > 100000 nM T67710 C6GAF5 155555773 IC50 = 4000 nM T67710 CFNP14 155557308 IC50 = 45000 nM T67710 CHDB02 155558265 IC50 = 23000 nM T67710 CGVN45 155559611 IC50 = 180 nM T67710 CTQ3H1 155560902 IC50 = 16000 nM T67710 C4DQ3V 155567876 EC50 > 100000 nM T68698 D0H1OL 135398635 Ki = 1472000 nM T68698 D0I7BL 65269 Ki = 110 nM T68698 D0I7TN 23190 IC50 = 4000 nM T68698 D0R2QS 72968 IC50 = 0.004 ug.mL-1 T68698 CY1P2C 72501 Ki = 4 nM T68698 CRG3J6 73651 Ki = 12 nM T68698 CI8KD2 97627 Ki = 410 nM T68698 C2CG8M 98567 Ki = 1930 nM T68698 CGF69C 99920 Ki = 3.3 nM T68698 C3BU7T 147104 Ki = 110 nM T68698 CHT80Q 275945 Ki = 22000 nM T68698 C8I2PG 358177 IC50 = 31 nM T68698 C3J5VD 402194 IC50 < 20000 nM T68698 CRU2Q9 443234 Ki = 39 nM T68698 CVQW71 451935 IC50 = 1000 nM T68698 C72EKO 469184 IC50 = 7600 nM T68698 CY0ZN2 472632 IC50 = 0.2 ug.mL-1 T68698 CA2U7Y 472655 IC50 > 10 ug.mL-1 T68698 C67BXW 481083 IC50 > 10 ug.mL-1 T68698 CJL5D2 489877 IC50 = 0.87 ug.mL-1 T68698 CLRY91 489878 IC50 = 3760 nM T68698 CLO12U 490351 Ki = 41 nM T68698 CJ2L8F 490432 IC50 = 123000 nM T68698 C5L8GI 490433 IC50 = 76000 nM T68698 CE9J3U 501516 Ki = 5020 nM T68698 C58AMW 501517 Ki = 27 nM T68698 CHNA61 501518 Ki = 586 nM T68698 C12AIT 501519 Ki = 22 nM T68698 C8T0YV 501520 Ki = 67600 nM T68698 CB4HR1 512554 IC50 > 10 ug.mL-1 T68698 CKIL63 512555 IC50 = 195 nM T68698 CTF70X 512656 IC50 > 10 ug.mL-1 T68698 CL24RG 512657 IC50 > 10 ug.mL-1 T68698 C1AU9I 512658 IC50 > 10 ug.mL-1 T68698 CL74IO 1362195 Ki = 1700 nM T68698 C13DGU 5358592 IC50 = 40 nM T68698 COLD86 6439007 Ki = 330 nM T68698 CX58IU 6450949 Ki = 125 nM T68698 CSB29R 6474190 IC50 = 90700 nM T68698 CW7NE1 6476927 IC50 = 8 nM T68698 CZR3N8 9816781 IC50 = 75020 nM T68698 CB01OK 9840103 Ki = 16000 nM T68698 CRAI41 9993207 Ki = 7900 nM T68698 C2SKW5 9997450 Ki = 134 nM T68698 CW21OU 10015023 IC50 = 7670 nM T68698 C3DI6E 10061387 Ki = 39 nM T68698 C4VB3K 10243225 Ki = 8800 nM T68698 CHG3J9 10400519 Ki = 273 nM T68698 C2FV5L 10422910 IC50 = 18 nM T68698 CNR64H 10655770 IC50 = 930 nM T68698 CR6A7V 11380460 IC50 = 12680 nM T68698 CJ8QH3 11537088 Ki = 17000 nM T68698 CV0F5A 11564784 Ki = 500 nM T68698 CTMK84 11615884 IC50 > 100000 nM T68698 CXEG94 11777524 Ki = 4500 nM T68698 C2RE5C 11779405 Ki = 110 nM T68698 CX35EZ 12097487 IC50 = 36460 nM T68698 C6IX0V 12769724 IC50 = 100000 nM T68698 C4SD3B 13712019 IC50 = 28000 nM T68698 CEC2K8 13939857 Ki = 35 nM T68698 CW0E2J 14134370 Ki = 160 nM T68698 CU06ED 14134371 IC50 = 1230 nM T68698 CB35KG 14134372 Ki = 200 nM T68698 C45LBI 14134395 IC50 = 950 nM T68698 CF9SO7 14134396 Ki = 200 nM T68698 CPJ92T 14134397 Ki = 170 nM T68698 C5YGX9 14134400 Ki = 90 nM T68698 CYGP51 14134401 Ki = 166 nM T68698 CCF8Z2 14134506 IC50 = 80 nM T68698 CFRL70 16075366 IC50 = 180 nM T68698 CZ03BO 21152084 Ki = 43400 nM T68698 CY07FB 25244925 Ki = 2600 nM T68698 C97ZIN 44189703 IC50 = 1.5 nM T68698 CL4K0U 44278585 Ki = 0.5 nM T68698 CYP2V1 44373339 IC50 > 100000 nM T68698 CS4NG1 44396071 IC50 > 100000 nM T68698 C7ZMI0 44396095 IC50 > 100000 nM T68698 C6BN5P 44396175 IC50 = 97270 nM T68698 CCW9P4 44432644 IC50 = 28940 nM T68698 CS2EY3 44450578 IC50 = 163000 nM T68698 C5JM9A 44450579 IC50 > 500000 nM T68698 CNI6X4 44451567 IC50 = 47200 nM T68698 CI3VJ8 44551468 IC50 = 400 nM T68698 CT8I2H 44561305 Ki = 12400 nM T68698 CVS3O8 44561306 Ki = 20300 nM T68698 C6BG4W 45110892 IC50 = 2.2 nM T68698 C7GN9D 45110893 IC50 = 36 nM T68698 CB5IQ2 45110895 IC50 = 98 nM T68698 CG5RZ9 45111029 IC50 = 4827 nM T68698 C5H3VJ 45111030 IC50 = 189 nM T68698 C36LBT 45111031 IC50 = 9.4 nM T68698 C50EYM 45111032 IC50 = 41 nM T68698 CJA7Q8 45111033 IC50 = 2.7 nM T68698 CL8NW5 45111034 IC50 = 1223 nM T68698 CYAQ84 45111036 IC50 = 28 nM T68698 C7RM9B 46174640 IC50 = 1.3 nM T68698 CZL10R 46874055 Ki = 94.6 nM T68698 CXH9E4 46874068 Ki = 4000 nM T68698 CY41AR 46874106 Ki = 67000 nM T68698 C3DB1E 46874218 Ki = 3100 nM T68698 CN59VL 46874243 Ki = 681 nM T68698 C0HY4G 46874757 Ki = 111 nM T68698 CS32QG 46874759 Ki = 101 nM T68698 C3F2PG 46874761 Ki = 10000 nM T68698 C0NLW6 46875043 Ki = 13700 nM T68698 C0DI9E 46875054 Ki = 45000 nM T68698 CD3C8F 46875063 Ki = 16000 nM T68698 CMGN58 46875065 Ki = 10000 nM T68698 CD28UB 46875621 Ki = 1100 nM T68698 CPHC63 46875632 Ki = 1700 nM T68698 CJ6EL3 46875710 Ki = 770 nM T68698 C19BFH 46875728 Ki = 48500 nM T68698 CE5O4A 46875732 Ki = 570 nM T68698 C8T2JI 46875733 Ki = 710 nM T68698 C7B8QH 46875922 Ki = 3600 nM T68698 CCE7X6 46875931 Ki = 3900 nM T68698 C2VZR9 46876033 Ki = 1300 nM T68698 CGJ03W 46876073 Ki = 96 nM T68698 CZ50WH 46876160 Ki = 3800 nM T68698 CY4L3V 46876365 Ki = 360 nM T68698 CTV70J 46876373 Ki = 570 nM T68698 CKB03R 46876407 Ki = 320 nM T68698 CH81PT 46877209 Ki = 75000 nM T68698 C5NFH6 46877212 Ki = 50000 nM T68698 C1O4WI 46877256 Ki = 750000 nM T68698 CWM2L0 46877257 Ki = 3200 nM T68698 C8IWQ3 46877302 Ki = 105000 nM T68698 CLG04P 46877303 Ki = 19000 nM T68698 C81YJV 46877310 Ki = 550 nM T68698 CJ23FN 46877328 Ki = 4000 nM T68698 CKE16H 46877337 Ki = 118500 nM T68698 CM4CG5 46877338 Ki = 96000 nM T68698 C0HQ5A 46877339 Ki = 17000 nM T68698 C6IRP9 46886640 IC50 > 250000 nM T68698 CW0Y4H 49797674 Ki = 19800 nM T68698 C8GU9B 51003093 IC50 = 60170 nM T68698 CM8WE3 51003094 IC50 > 1000000 nM T68698 C7M3KT 51003095 IC50 > 1000000 nM T68698 C46DIL 51003096 IC50 > 1000000 nM T68698 CZK6B3 53318848 IC50 > 1000000 nM T68698 CC6GR8 57522307 IC50 = 910 nM T68698 C0Z8LK 68364288 IC50 = 2300 nM T68698 CIX13E 73351185 Ki = 1900 nM T68698 C8H9WC 73352895 Ki = 800 nM T68698 CPHB93 90644119 IC50 > 10000 nM T68698 CWP2F5 90644120 IC50 = 2100 nM T68698 C28IXS 90644121 IC50 > 10000 nM T68698 C8INM3 90644122 IC50 = 672 nM T68698 C7ZQA6 90644123 IC50 = 878 nM T68698 C4Y6KI 90644124 IC50 = 1960 nM T68698 CD2X0B 90644125 IC50 = 976 nM T68698 CS3KR7 91824125 Ki = 1.5 nM T68698 C4F3MG 118710205 IC50 = 530 nM T68698 C1PIQ5 118710206 IC50 = 380 nM T68698 C6TMO4 118710207 IC50 = 340 nM T68698 C7IDP1 118710208 IC50 = 970 nM T68698 CG5M1W 118710209 IC50 = 8780 nM T68698 CN29AS 118710210 IC50 = 11360 nM T68698 C0RW1F 118710211 IC50 > 100000 nM T68698 C87EMG 118710212 IC50 = 17000 nM T68698 CMWO70 118710213 IC50 = 2700 nM T68698 C39PRU 118710214 IC50 = 52 nM T68698 CT9PF2 118710215 IC50 = 81 nM T68698 CV51BZ 118710216 IC50 = 530 nM T68698 C5YR2F 118710217 IC50 > 100000 nM T68698 CGT1A9 118710218 IC50 = 4600 nM T68698 CM64LA 118710219 IC50 = 230 nM T68698 CKP9S8 118710220 IC50 = 890 nM T68698 CBW08J 118710221 IC50 = 13 nM T68698 CLAB80 118710222 IC50 = 200 nM T68698 CD01LY 118710223 IC50 = 49 nM T68698 C7HJ8B 118710224 IC50 = 44 nM T68698 C5J7EQ 118710225 IC50 = 330 nM T68698 C01AOB 118710226 IC50 = 320 nM T68698 COMR26 118710227 IC50 = 130 nM T68698 C3AY7W 118710228 IC50 = 70 nM T68698 C91TJV 118710229 IC50 = 60 nM T68698 C1S0YD 118710230 IC50 = 49 nM T68698 C29JSZ 118710231 IC50 = 1200 nM T68698 CI8Z4P 118710232 IC50 = 1500 nM T68698 C34ARU 118710233 IC50 = 110 nM T68698 CR26QJ 118710234 IC50 = 600 nM T68698 CVL4C5 118710235 IC50 = 150 nM T68698 CEW89M 118718118 Ki = 224 nM T68698 CY4DU7 122178501 IC50 > 100000 nM T68698 CGY0N1 122178503 IC50 > 100000 nM T68698 CD98QW 122178504 IC50 > 100000 nM T68698 CX8FW7 122178506 IC50 > 100000 nM T68698 CA98UV 122183895 IC50 = 640 nM T68698 CQ0LA3 122183896 IC50 > 100000 nM T68698 CK6J3X 122183897 IC50 > 100000 nM T68698 CNOV-65 122183898 IC50 = 70 nM T68698 CQM0H1 122183899 IC50 = 60 nM T68698 C6JAU8 122183900 IC50 = 49 nM T68698 CMU94S 122183901 IC50 = 1200 nM T68698 CTU42V 122183902 IC50 = 1500 nM T68698 C0SZO2 122183903 IC50 = 110 nM T68698 CHM13L 122183904 IC50 = 600 nM T68698 C80TRM 122183905 IC50 = 150 nM T68698 CI8WG9 122183915 IC50 = 8.5 nM T68698 CP1FW4 135398641 Ki = 925000 nM T68698 CP4M0E 135976391 Ki 128000 nM T68698 C8WD3Z 135976393 Ki = 422000 nM T68698 CZD50N 137090971 IC50 > 100000 nM T68698 CJW84E 137090972 IC50 > 100000 nM T68698 C5ZM8O 137628302 IC50 > 10000 nM T68698 CW0C4P 155517779 IC50 > 3700 nM T68698 CNP67J 155524359 IC50 > 100000 nM T68698 CKN0W4 155530574 IC50 > 100000 nM T68698 CI2OR3 155531848 IC50 = 4390 nM T68698 CAE5R9 155536819 IC50 > 100000 nM T68698 CZXU90 155538219 IC50 > 100000 nM T68698 CTM53Z 155543643 IC50 > 100000 nM T68698 CKWS45 155544569 IC50 > 100000 nM T68698 CDU83I 155549525 IC50 = 760 nM T68698 CKP82O 155553203 IC50 = 1060 nM T68698 C09CGT 155568198 IC50 > 100000 nM T68698 C0I9OP 155568822 IC50 > 100000 nM T68698 D02XPR 73124 IC50 = 280 nM T68698 D02YYQ 23661679 IC50 = 7530 nM T68698 D0D2MS 11737492 IC50 = 15700 nM T68698 D0F5AJ 126704 Ki = 160 nM T68698 D0O2CM 498018 IC50 = 480 nM T68698 D0X3MK 73087 IC50 = 440 nM T04689 D0T8GD 89594 EC50 = 180000 nM T04689 D09ADT 119380 EC50 = 411000 nM T04689 CUI25G 115224 IC50 = 120000 nM T04689 CY1XN7 7446712 IC50 = 1000 nM T04689 C74CBS 9794141 EC50 = 34000 nM T04689 C0Z5RS 9859386 IC50 = 6000 nM T04689 CLWT60 9882021 EC50 > 100000 nM T04689 CDH4J3 10130527 IC50 = 11000 nM T04689 C6LB2N 10130752 IC50 = 8000 nM T04689 CIQ12L 11701287 Ki = 944 nM T04689 CY7F5O 15389735 EC50 > 1000000 nM T04689 CQ03LX 21290600 IC50 = 81000 nM T04689 CW2R4M 23624283 IC50 = 3981.07 nM T04689 CC1SF7 49863118 IC50 = 794.33 nM T04689 CJ34EQ 53483935 IC50 = 4200 nM T04689 CLH24J 56663402 IC50 > 10000 nM T04689 CU7OP3 56666825 IC50 > 10000 nM T04689 CY01LS 56666826 IC50 > 10000 nM T04689 CCP40B 56666827 IC50 > 10000 nM T04689 CVT85Q 56670262 IC50 = 7800 nM T04689 C7XK8I 56677105 IC50 = 5500 nM T04689 C02AZR 56677106 IC50 > 10000 nM T04689 CL45WN 57345320 IC50 > 30000 nM T04689 CV2J9A 57663655 IC50 = 6309.57 nM T04689 CU3D9N 73388373 EC50 = 19952.62 nM T04689 CI14LP 145949343 IC50 = 11300 nM T04689 CGW92C 145952721 IC50 > 30000 nM T04689 D0R4RN 1204 IC50 = 160 nM T33966 CSD1A3 125874 Ki = 200 nM T33966 CX7U8V 444797 Ki = 450 nM T33966 CF5A3T 9837547 IC50 > 50000 nM T33966 CHI95J 9926432 IC50 = 1400 nM T33966 CM1A0D 9943447 IC50 = 6400 nM T33966 CVK4L6 10418061 IC50 = 3900 nM T33966 C6FQ0R 10465893 IC50 = 1700 nM T33966 CT7IR8 12110710 IC50 > 100000 nM T33966 CFQW82 18955956 Ki = 207000 nM T33966 CYT07N 21575382 IC50 = 0.007 ug.mL-1 T33966 CG0M4T 21575383 IC50 = 3.4 ug.mL-1 T33966 C4UDA1 21606664 IC50 = 0.0052 ug.mL-1 T33966 CR1BW2 21606665 IC50 = 0.0076 ug.mL-1 T33966 C14ZMJ 24768537 Ki = 150 nM T33966 C7J1DP 24774575 Ki = 15000 nM T33966 CP2LY7 25033280 Ki = 17000 nM T33966 C4YKQ1 25033281 Ki = 22000 nM T33966 CA9D6R 25209871 IC50 = 0.12 ug.mL-1 T33966 C46SPD 44374719 Ki = 6500 nM T33966 C0NI9F 44374736 Ki = 5820 nM T33966 CFPX72 44374737 Ki = 4950 nM T33966 CPRQ07 44374750 Ki = 1200 nM T33966 C9RPC6 44374765 Ki = 1160 nM T33966 C1CPB2 44374994 Ki = 980 nM T33966 CXTF63 44374995 Ki = 560 nM T33966 CGD91Y 44374996 Ki = 5900 nM T33966 C4UBK7 44374998 Ki = 320 nM T33966 CG75AN 44377126 Ki = 1200 nM T33966 C6SV1C 44387258 IC50 = 1100 nM T33966 C06HJB 44446952 Ki = 11000 nM T33966 CNK7X5 44446953 Ki = 35000 nM T33966 CEB78N 44446954 Ki = 11000 nM T33966 CMO78A 44446956 Ki = 530 nM T33966 CV6H2M 44446957 Ki = 350 nM T33966 CF4KE1 44446959 Ki = 3600 nM T33966 CW9C0E 44446960 Ki = 7200 nM T33966 CQB5M0 44446963 Ki = 9900 nM T33966 C94POY 44446965 Ki = 5000 nM T33966 CBX2U9 44446967 Ki = 2300 nM T33966 CRZ6B3 44446968 Ki = 14000 nM T33966 CY9O4I 44446969 Ki = 8900 nM T33966 C4PQ7D 44446970 Ki = 1600 nM T33966 C96KIY 44446972 Ki = 5000 nM T33966 CK1EM5 44446974 Ki = 4600 nM T33966 C4V6RZ 44446975 Ki = 16000 nM T33966 CBL9E6 44446976 Ki = 1900 nM T33966 CVYX54 44446979 Ki = 3300 nM T33966 CAI9Z6 44446980 Ki = 4600 nM T33966 C86KVP 44446984 Ki = 11000 nM T33966 CYQN96 44452011 Ki = 2080 nM T33966 CFOM52 44452012 Ki = 790 nM T33966 CJ8G5P 44452013 Ki = 68000 nM T33966 CZI4H9 44452015 Ki = 62600 nM T33966 CC2IS3 44454957 Ki = 12000 nM T33966 C1ESI2 44454959 Ki = 12000 nM T33966 C8L0MV 44454960 Ki = 12000 nM T33966 CBG6T0 44454987 Ki = 15000 nM T33966 CN7UW3 44455013 Ki = 8900 nM T33966 CC5L7S 44455015 Ki > 50000 nM T33966 C6KDT1 44455016 Ki = 9300 nM T33966 CF4ML7 44455018 Ki = 14000 nM T33966 CZI6S1 44455047 Ki = 1700 nM T33966 C3UF6E 44455406 Ki = 5000 nM T33966 CJG71N 44455407 Ki = 32000 nM T33966 C0IR5W 44455428 Ki = 17000 nM T33966 C62KSV 44455429 Ki > 50000 nM T33966 CR9WL2 44455430 Ki = 11000 nM T33966 CXD0Q4 44558923 IC50 = 0.022 ug.mL-1 T33966 C48QBD 45101440 Ki = 160 nM T33966 CP43WZ 45484707 Ki = 430 nM T33966 C2Q9OC 45484717 Ki = 31000 nM T33966 C85MBH 112499885 Ki = 0.087 nM T33966 C2L8SI 112499886 Ki = 0.107 nM T33966 CS49EB 112499887 Ki = 0.04 nM T33966 CG9SC3 145949929 Ki = 289000 nM T33966 C8H1FK 145950532 Ki = 294000 nM T33966 CH02KU 145955234 Ki = 56000 nM T33966 CA6QF8 145956086 Ki = 413000 nM T33966 CZH6P7 145956217 Ki = 238000 nM T33966 CF01VH 145974566 Ki = 60400 nM T33966 CU65CB 155511784 Ki = 0.08 nM T33966 CFG96J 155514645 Ki = 5.9 nM T33966 CF64GH 155518335 Ki = 0.07 nM T33966 CY0H2S 155519530 Ki = 3.1 nM T33966 CA49SR 155523686 Ki = 1.7 nM T33966 C5X4TD 155524117 Ki = 0.1287 nM T33966 C4F1EB 155538870 Ki = 0.3 nM T33966 CD81NB 155547411 Ki = 1.2 nM T33966 D06LNX 3858 IC50 = 400 nM T33966 D0N4RO 44377139 Ki = 310 nM T06792 D00UVA 11556711 IC50 = 2420 nM T06792 D0SH3I 387447 IC50 = 3 nM T06792 D0DP0J 92135659 IC50 = 1840 nM T06792 D0VO0T 24800541 IC50 = 1 nM T06792 CLU69K 10628969 IC50 = 440 nM T06792 CU0FE7 24752894 IC50 = 104 nM T06792 CN62YJ 46850523 IC50 = 140 nM T06792 CEV5D1 49859748 IC50 = 10600 nM T06792 C3QG8L 59127842 IC50 = 36 nM T06792 C82JTA 71305068 IC50 = 21500 nM T06792 C45HOE 71562349 IC50 > 10000 nM T06792 CGY43C 78425867 IC50 = 1850 nM T06792 CC0OF1 101874274 IC50 = 300 nM T06792 CG0N1O 101874275 IC50 = 7100 nM T06792 CL50TR 101874276 IC50 = 7300 nM T06792 C0RY3V 101874277 IC50 = 6200 nM T06792 CVHC29 101874278 IC50 > 100000 nM T06792 C4VHU6 101874279 IC50 > 100000 nM T06792 C9C5OZ 117607839 IC50 = 3530 nM T06792 CLHS74 117607901 IC50 = 223 nM T06792 CW9R0U 117607904 IC50 = 0.623 nM T06792 C7QST8 117611788 IC50 = 51 nM T06792 CO1HJ9 117611880 IC50 = 140 nM T06792 C9YH1X 117611941 IC50 = 112 nM T06792 CO6E0B 118709670 IC50 = 170 nM T06792 C8WMH3 118709671 IC50 = 68 nM T06792 CZ8GE0 118709672 IC50 = 96 nM T06792 CZ70XF 118709673 IC50 = 67 nM T06792 C7C9PZ 118709674 IC50 = 220 nM T06792 CS05KF 118709675 IC50 = 22 nM T06792 C17ZTF 118709676 IC50 = 34 nM T06792 C0WZ3V 118709677 IC50 = 66 nM T06792 C14VLB 118709678 IC50 = 87 nM T06792 CO5CU1 118709679 IC50 = 42 nM T06792 C1RA9C 118709680 IC50 = 130 nM T06792 C9BWP4 145979302 IC50 = 5700 nM T06792 CN79HG 145979487 IC50 = 3500 nM T06792 CEI3U1 145979850 IC50 = 4800 nM T06792 CG6UL0 145980995 IC50 = 4000 nM T06792 CB67YT 145981691 IC50 = 16100 nM T06792 C41IRV 145981707 IC50 = 14000 nM T06792 CL1F8N 145982922 IC50 = 13000 nM T06792 C5X3GQ 145986425 IC50 = 12600 nM T06792 CRZE86 145986857 IC50 = 45000 nM T06792 CHWT73 145987085 IC50 = 8900 nM T06792 CM3H4F 145987197 IC50 = 4300 nM T06792 CNZ7R6 145987536 IC50 = 12500 nM T06792 C1EF3B 145988020 IC50 = 23800 nM T06792 CQIS01 145988427 IC50 = 7310 nM T06792 CE16JH 145989568 IC50 = 52000 nM T06792 CXG30R 145990249 IC50 = 21000 nM T06792 C8IL9E 145992200 IC50 = 10320 nM T06792 CBY18W 145992498 IC50 = 2770 nM T06792 C6GHQ9 145993211 IC50 = 59000 nM T06792 CEVY70 145993649 IC50 = 24600 nM T06792 CJO08K 145993925 IC50 = 8800 nM T06792 C8E6ZX 155514792 IC50 > 10000 nM T06792 CX76LO 155515463 IC50 > 10000 nM T06792 C53ZEN 155516179 IC50 > 100000 nM T06792 CM3BV8 155516620 IC50 > 100000 nM T06792 CE95IQ 155518158 IC50 > 100000 nM T06792 CNM0Q9 155521286 IC50 > 100000 nM T06792 CZKF54 155521690 IC50 > 10000 nM T06792 CB0WG8 155522381 IC50 = 743.5 nM T06792 C8GNQ9 155522828 IC50 > 25000 nM T06792 CW75YK 155523151 IC50 > 100000 nM T06792 CAC34Y 155527225 IC50 = 3100 nM T06792 CUP2B4 155531358 IC50 = 415 nM T06792 C2NTI6 155538936 IC50 > 100000 nM T06792 C6OIY3 155541618 IC50 > 100000 nM T06792 C12LPX 155551071 IC50 > 10000 nM T06792 CBHM14 155553205 IC50 > 100000 nM T06792 C35NJC 155553210 IC50 > 10000 nM T06792 CI15FC 155553565 IC50 > 10000 nM T06792 CVJ3E7 155553910 IC50 > 100000 nM T06792 C6YP0L 155554916 IC50 > 100000 nM T06792 C5Z7YC 155567712 IC50 > 10000 nM T06792 C4ZV3Q 155568941 IC50 > 10000 nM T06792 D0Q4MO 23642227 IC50 = 287 nM T01943 D04AIT 5280445 IC50 = 5000 nM T01943 D0K8KX 5280343 IC50 = 1500 nM T01943 D0L4FS 5280961 IC50 = 7000 nM T01943 D0U2BH 65064 IC50 = 400 nM T01943 CY0AL9 72279 IC50 = 30000 nM T01943 CNIW58 107905 IC50 = 400 nM T01943 CDZ65K 199472 IC50 = 600 nM T01943 CN7AQ6 15958429 IC50 = 14 ug.mL-1 T01943 CZR73C 16072317 IC50 = 12.5 ug.mL-1 T01943 C20YLR 22600366 IC50 = 0.58 ug.mL-1 T01943 C15VRN 44412009 IC50 = 40000 nM T01943 C6XHE9 49770727 IC50 = 12 ug.mL-1 T01943 CG4H0W 71768351 IC50 > 100000 nM T01943 CMAP17 71768352 IC50 = 16300 nM T01943 CW0T6G 72703050 IC50 > 100000 nM T01943 CPZO91 72703242 IC50 > 100000 nM T01943 CQ2IU6 72703243 IC50 = 90000 nM T01943 C0B3KS 72703244 IC50 = 13000 nM T01943 CE6HI7 72703245 IC50 = 28000 nM T01943 CJ12BK 72703246 IC50 = 10000 nM T01943 CESN04 73347724 IC50 > 100000 nM T01943 D01KKU 5281894 IC50 = 20000 nM T01943 D02TVS 985 IC50 > 100 ug.mL-1 T01943 D0MF5Y 5281614 IC50 = 2000 nM T01943 D0NJ4H 5281670 IC50 = 8000 nM T01943 D0RB1V 6419835 IC50 = 400 nM T01943 D0S9YX 5280373 IC50 = 8000 nM T01943 D0SY2M 5281708 IC50 = 30000 nM T01943 D0T3PW 5281672 IC50 = 2000 nM T19229 D01KKQ 135400182 IC50 = 99.5 nM T19229 D02LWU 148121 IC50 = 57 nM T19229 D0SV8E 126941 IC50 = 121 nM T19229 D0Y4GO 135410875 IC50 = 13.2 nM T19229 CPM3L5 67092576 IC50 > 1000 nM T19229 CTK64O 67092918 IC50 > 1000 nM T19229 C87FBU 135455948 IC50 = 80.2 nM T19229 CF8D5O 135465664 IC50 > 1000 nM T19229 C9Z4ES 135567027 IC50 = 5.21 nM T19229 C14LTO 135567028 IC50 = 43.4 nM T19229 CF39AI 135567029 IC50 = 3.34 nM T19229 C8N7ES 135567030 IC50 = 41.5 nM T19229 CGM2V5 135567031 Ki = 420 nM T19229 CFE2O7 135567034 IC50 = 40 nM T19229 C8KVP5 135567035 IC50 = 6.51 nM T19229 CSQX75 135567163 IC50 = 87.4 nM T19229 CQF8P5 135800109 IC50 = 9.71 nM T19229 C6XK3M 135862924 Ki = 100 nM T19229 CL8VN5 136015502 IC50 = 312 nM T19229 CR7UY3 136044173 IC50 > 1000 nM T19229 C0Q5FI 136044174 IC50 > 1000 nM T19229 CGX68Y 136044175 IC50 > 1000 nM T19229 C4C9FN 136044176 IC50 > 1000 nM T19229 CIPD35 136044177 IC50 > 1000 nM T19229 CZG8W6 136059167 IC50 = 30.4 nM T19229 CZC95Y 136059168 IC50 > 1000 nM T19229 CG2ID9 136059169 IC50 > 1000 nM T19229 C2WH0S 136059178 IC50 > 1000 nM T19229 CB3GL7 136059191 IC50 > 1000 nM T19229 CCHG08 136059192 IC50 > 1000 nM T19229 C4Q1HF 136180345 IC50 = 141 nM T19229 CDC83K 136180346 IC50 = 57.4 nM T19229 CF7NW6 136180347 IC50 > 1000 nM T19229 CPH52E 137150145 IC50 > 1000 nM T19229 C9XD1M 137150146 IC50 = 747 nM T19229 CHDB56 137150160 IC50 = 48.6 nM T19229 CUF8R1 155515541 IC50 = 207 nM T19229 CMKA64 155517044 IC50 = 81.7 nM T19229 CCL3Y9 155518053 IC50 = 20.4 nM T19229 C91SVN 155519837 IC50 = 57.5 nM T19229 CO7BN6 155524531 IC50 > 1000 nM T19229 CT70WU 155530762 IC50 = 5.01 nM T19229 CX42MF 155532591 IC50 = 267 nM T19229 CFU98A 155534971 IC50 = 88.5 nM T19229 C4K2RU 155538415 IC50 > 1000 nM T19229 C27BIX 155539477 IC50 > 1000 nM T19229 C6S7OC 155548982 IC50 = 3.82 nM T19229 CX3K8F 155549935 IC50 = 4.57 nM T19229 CJ0MK5 155554671 IC50 = 67 nM T19229 CYQ0I9 155555353 IC50 = 109 nM T90987 CJS23I 9868333 Ki = 7800 nM T90987 CY08WJ 10322755 Ki = 7800 nM T90987 C8C5AV 11294179 Ki > 1000 nM T90987 CZB81D 44395506 IC50 = 79 nM T90987 C52ESR 66559934 IC50 > 50000 nM T90987 C57ARI 66560021 IC50 > 50000 nM T90987 CU58DB 66560022 IC50 > 50000 nM T90987 C16RDM 66560389 IC50 > 50000 nM T90987 C8RZG9 66560479 IC50 > 50000 nM T90987 CKW2Q5 71453375 IC50 > 50000 nM T90987 D0H6CK 10160968 Ki = 776 nM T06569 D00STL 644241 Ki = 461 nM T06569 D01MUR 68844 Ki = 0.9 nM T06569 D02PJA 24841 Ki = 810000 nM T06569 D03QGM 5355 Ki = 0.8 nM T06569 D03RTS 2662 Ki = 94 nM T06569 D03UOT 785 Ki = 521000 nM T06569 D05OFX 219078 Ki = 412 nM T06569 D05UYW 5284549 Ki = 10 nM T06569 D07HBX 338 Ki = 11900 nM T06569 D07INV 3295 Ki = 43 nM T06569 D07VDZ 5284627 Ki = 45 nM T06569 D09NIA 2732 Ki = 1347 nM T06569 D09VAZ 5565 Ki = 43000 nM T06569 D0AZ3C 5291 Ki = 392 nM T06569 D0AZ8C 5213 Ki = 9700 nM T06569 D0C2II 4100 Ki = 10 nM T06569 D0C8FX 3005837 Ki = 2410 nM T06569 D0E1SW 1986 Ki = 11 nM T06569 D0H8FH 3702 Ki = 1606 nM T06569 D0J4GO 3038 Ki = 79 nM T06569 D0J7RK 36811 Ki = 9470 nM T06569 D0K0OZ 5702160 Ki = 98.2 nM T06569 D0K1QD 3998 Ki = 4800 nM T06569 D0K8KX 5280343 Ki = 6170 nM T06569 D0L4JT 5333 Ki = 941 nM T06569 D0L6DA 119607 Ki = 572 nM T06569 D0OT0O 44561 Ki = 1810000 nM T06569 D0PQ3G 3440 Ki = 245 nM T06569 D0SH3I 387447 Ki = 4380 nM T06569 D0U5QK 1983 Ki = 658000 nM T06569 D0Y2IZ 5560 Ki = 2459 nM T06569 D0Z3EI 6038 Ki = 33 nM T06569 D04IIU 216468 Ki = 47 nM T06569 D05NJI 5287541 Ki = 653 nM T06569 D06PII 5356 Ki = 134 nM T06569 D08BXT 1102 Ki = 1410 nM T06569 D0L6HN 996 Ki = 208000 nM T06569 D0U3EP 445154 Ki = 8070 nM T06569 D0V0UK 82267 Ki = 0.07 nM T06569 D03SLR 445858 Ki = 8450 nM T06569 D0NH9P 135 Ki = 5700 nM T06569 D0LD9S 1103 Ki = 990 nM T06569 CI0WH9 72 Ki = 4720 nM T06569 CUT2V4 260 Ki = 730000 nM T06569 COV5W3 402 Ki = 710000 nM T06569 CSZ43B 540 Ki = 690000 nM T06569 C97QXH 767 Ki = 690000 nM T06569 C39CTO 768 Ki = 70000 nM T06569 C1QDT0 781 Ki = 890000 nM T06569 CAD4R0 798 Ki = 3630 nM T06569 CW0R2L 944 Ki = 760000 nM T06569 CQV86E 1100 Ki = 14200000 nM T06569 C8W7BZ 1118 Ki = 9900000 nM T06569 CU12QE 1203 Ki = 4910 nM T06569 C5L7VX 2871 Ki = 2230 nM T06569 CJ2F6P 5056 Ki = 8630 nM T06569 CDJ4K6 5987 Ki = 0.09 nM T06569 CUP2F4 7043 Ki = 234700 nM T06569 C1CVT7 7121 Ki = 24420 nM T06569 C6NC4O 7414 Ki = 5100 nM T06569 CJKY76 7420 Ki = 3170 nM T06569 CIU0C8 7519 Ki = 234700 nM T06569 CUG8B9 11418 Ki = 402300 nM T06569 CCPT31 11419 Ki = 427100 nM T06569 CUA0L6 14917 Ki = 600000 nM T06569 C3NG2U 24529 Ki = 820000 nM T06569 CFM9L6 24530 Ki = 70000 nM T06569 C4OU6D 35703 Ki = 82300 nM T06569 C1N6SE 61127 Ki = 29138 nM T06569 CE5RZ1 76509 Ki = 780 nM T06569 CX47BZ 78479 Ki = 53000 nM T06569 CEC01M 97598 Ki = 12840 nM T06569 CN19UT 129695 Ki = 110 nM T06569 CUX39B 132037 Ki = 3410 nM T06569 CVB67D 134560 Ki = 73 nM T06569 CD2HC7 138614 Ki = 405600 nM T06569 C8AO0Z 165323 Ki = 114 nM T06569 C1QOB5 284045 Ki = 382473 nM T06569 CT3ZU4 388776 Ki = 1100 nM T06569 CH21KA 389641 Ki = 104000 nM T06569 C6CQO3 389642 Ki = 114000 nM T06569 CNPZ40 394897 Ki = 765 nM T06569 C4TD8M 2388085 Ki > 10000 nM T06569 C21FUI 2801263 Ki = 3790 nM T06569 CE2GR3 2900806 Ki = 109000 nM T06569 CI8JY0 5172475 Ki = 740 nM T06569 C9L8AX 6537802 Ki = 41 nM T06569 C65FRB 6852128 Ki = 136 nM T06569 CKCM96 7463376 Ki = 8580 nM T06569 CDCP43 7766335 Ki = 420 nM T06569 CY47OI 9998322 Ki = 24 nM T06569 CWM01R 10059806 Ki = 13692 nM T06569 CD58EL 10083644 Ki = 730 nM T06569 C58IYR 10366827 Ki = 590 nM T06569 C3HBY6 10375558 Ki = 4150 nM T06569 C73KXU 10586607 Ki = 6700 nM T06569 C9TSQ6 10632698 Ki = 43100 nM T06569 C8C6ER 11069133 Ki = 41 nM T06569 C39IDU 11183936 Ki = 12010 nM T06569 CHC42Y 11245700 Ki = 654 nM T06569 CA6T0Z 11322287 Ki = 11660 nM T06569 CXB86F 11579563 Ki = 12530 nM T06569 CDU79V 11637531 Ki = 10820 nM T06569 CX4W3J 11701693 Ki = 9870 nM T06569 CV7HN1 11795548 Ki = 65 nM T06569 CMPA32 12066940 Ki > 500000 nM T06569 CB15KR 12066941 Ki > 500000 nM T06569 CREV05 12140130 Ki = 12430 nM T06569 CHOG93 14611919 Ki = 2650 nM T06569 C8PER5 15938557 Ki > 500000 nM T06569 CC0Z4V 16119626 Ki = 510 nM T06569 C6SFI8 18268734 Ki > 10000 nM T06569 C61KUX 21726402 Ki = 9680 nM T06569 C54IUM 21778115 Ki = 17830 nM T06569 C27BJH 21778117 Ki = 17430 nM T06569 C9U4TE 22313850 Ki = 1230 nM T06569 CICR37 23426698 Ki = 38190 nM T06569 CPN2T5 25392418 Ki > 10000 nM T06569 C82MRL 44144383 Ki = 25 nM T06569 CI3O9B 44395149 Ki = 147 nM T06569 CZ4DF9 44399462 Ki = 76 nM T06569 CD5MJ6 44399571 Ki = 59 nM T06569 C2T7MB 44399654 Ki = 749 nM T06569 C8E0MV 44552472 Ki = 9210 nM T06569 CKG53H 44552473 Ki = 1920 nM T06569 C17XAJ 44552559 Ki = 4170 nM T06569 CF0KQ8 44581932 Ki = 73 nM T06569 C23MVW 45269009 IC50 = 35700 nM T06569 C0RG8K 45269749 Ki > 100000 nM T06569 CV5RQ3 45484187 Ki = 4300 nM T06569 CTG20B 45485271 Ki = 100 nM T06569 CK4U0V 45485283 Ki = 5600 nM T06569 CHE08Y 46225608 Ki = 10230 nM T06569 CIE2H3 46225609 Ki = 9640 nM T06569 CF42NR 46225631 Ki = 7610 nM T06569 C0ZG3L 46225639 Ki = 7960 nM T06569 CGW1I5 46225644 Ki = 7840 nM T06569 CEOQ06 46225645 Ki = 8310 nM T06569 CR0WO3 46225646 Ki = 8540 nM T06569 CC2BL5 46225656 Ki = 8980 nM T06569 CW52PZ 46225672 Ki = 4950 nM T06569 CXJ1C9 46225673 Ki = 4310 nM T06569 C93AIR 46899573 Ki = 156000 nM T06569 CJ0R2O 46911381 Ki = 921 nM T06569 CF89ML 53307609 Ki = 29670 nM T06569 C0NUM6 53386724 Ki = 980 nM T06569 C54FGU 53386866 Ki = 543 nM T06569 CRI54V 53386867 Ki = 1035 nM T06569 CUX7S4 53386868 Ki = 814 nM T06569 CIJ9V0 56684131 Ki = 8140 nM T06569 CH52DA 56921864 Ki = 8950 nM T06569 CUR32K 57334711 Ki = 480 nM T06569 C2CD1R 57334712 Ki = 470 nM T06569 C1K0DM 57334713 Ki = 470 nM T06569 CP7YR5 57345662 Ki = 8 nM T06569 C13FJU 57392368 Ki = 510 nM T06569 CY5G4Z 57395885 Ki = 960 nM T06569 C5RX6H 57396029 Ki = 5240 nM T06569 CP75OF 57397664 Ki = 158592 nM T06569 CUAG84 57397836 Ki = 765300 nM T06569 CW43HV 57397837 Ki = 5590 nM T06569 C1MCW8 57399336 Ki = 919182 nM T06569 C2CAM1 57399491 Ki = 4810 nM T06569 C2J7GW 66572313 Ki = 35450 nM T06569 C7J5RN 66573254 Ki = 45360 nM T06569 CQR91N 70692438 Ki = 28170 nM T06569 CWJ0Q8 70696540 Ki = 11143 nM T06569 CXJ16H 71450117 Ki = 8055 nM T06569 CB8JA3 71455488 Ki = 9340 nM T06569 C02UHX 71455489 Ki = 7116 nM T06569 CICJ97 71457274 Ki = 9280 nM T06569 CMHG14 71521493 Ki = 6200 nM T06569 CHN53G 71521494 Ki = 7700 nM T06569 CZJ5M6 71521495 Ki = 7900 nM T06569 CFBE53 71521496 Ki > 100000 nM T06569 CME27W 71521497 Ki = 8100 nM T06569 C24XWU 71521575 Ki = 8800 nM T06569 CJF68W 71521576 Ki > 100000 nM T06569 CX82JD 72696463 Ki = 130 nM T06569 COCV73 72696591 Ki = 1388 nM T06569 C5KHD7 72696592 Ki = 220 nM T06569 C4FBA6 72696593 Ki = 274 nM T06569 CO1JM5 72696594 Ki = 167 nM T06569 CUF61Q 72696595 Ki = 148 nM T06569 CO1JT3 73054728 Ki = 857 nM T06569 CDGZ03 101879106 Ki > 120 nM T06569 CY6ER7 101879108 Ki > 120 nM T06569 C0D1SQ 118724328 Ki > 120 nM T06569 C89YTC 118724329 Ki > 120 nM T06569 CBT87C 118724330 Ki > 120 nM T06569 C49AWZ 118724331 Ki > 120 nM T06569 CH1N0C 122193189 Ki = 560 nM T06569 C19HVL 122193190 Ki = 740 nM T06569 C5TQJ1 122193251 Ki = 540 nM T06569 C8XCL0 122193252 Ki = 470 nM T06569 CIX41M 138393379 Ki > 10000 nM T06569 CBOM51 138753317 Ki > 10000 nM T06569 COP4Q6 155516517 Ki = 9192 nM T06569 CAG9L4 155517430 Ki = 2440 nM T06569 CP49HE 155520274 Ki = 7428 nM T06569 CTJ3I7 155530506 Ki = 7218 nM T06569 CT5NG1 155534179 Ki > 10000 nM T06569 CVU5P6 155535355 Ki > 10000 nM T06569 C8RV6T 155541805 Ki > 10000 nM T06569 CU1NE7 155549031 Ki > 10000 nM T06569 CWB82E 155555878 Ki > 10000 nM T06569 CH5VU6 155568899 Ki > 10000 nM T06569 D00IUB 13019 Ki = 13700 nM T06569 D00RNZ 910172 Ki = 93100 nM T06569 D00XJA 711717 Ki = 65200 nM T06569 D00YEF 148885 Ki = 1414 nM T06569 D01BUB 94952 Ki = 90600 nM T06569 D01STY 9861037 Ki = 1024 nM T06569 D02DBP 5054 Ki = 550000 nM T06569 D02QGI 273 Ki = 740 nM T06569 D03NBX 637308 Ki = 770 nM T06569 D03ZMQ 323 Ki = 2000 nM T06569 D04CVC 4687472 Ki = 96 nM T06569 D04NSN 169682 Ki = 813 nM T06569 D05QUG 45485279 Ki > 500000 nM T06569 D05TLB 11117301 Ki = 795 nM T06569 D05WQF 637540 Ki > 1000000 nM T06569 D05XZM 10081162 Ki = 6680 nM T06569 D06DYP 234562 Ki = 44500 nM T06569 D06TPF 1057 Ki = 520 nM T06569 D07MTM 403 Ki = 23500 nM T06569 D07QJJ 289 Ki = 606000 nM T06569 D07TAJ 914298 Ki = 6600 nM T06569 D09JPC 16402 Ki = 720 nM T06569 D09PWX 8739 Ki = 887 nM T06569 D09QHC 7370 Ki = 2970 nM T06569 D09WSJ 19772348 Ki = 1334 nM T06569 D09WVV 8111 Ki = 11500 nM T06569 D0A0YX 5143 Ki = 935 nM T06569 D0A1CM 5281855 Ki = 7060 nM T06569 D0A6HS 6852129 Ki = 103 nM T06569 D0AU0M 637542 Ki = 6720 nM T06569 D0C7LR 313 Ki = 720000 nM T06569 D0D4OV 20043772 Ki = 1020 nM T06569 D0D6UR 12394434 Ki > 500000 nM T06569 D0E8CC 18794 Ki = 93 nM T06569 D0EJ9B 66827 Ki = 0.82 nM T06569 D0G0FJ 11206245 Ki = 1090 nM T06569 D0G3BI 25090 Ki = 54700 nM T06569 D0H3NS 10752 Ki = 76300 nM T06569 D0L5TZ 20195365 Ki = 9300 nM T06569 D0LU4S 156219 Ki = 13000 nM T06569 D0M3PO 69561 Ki = 955 nM T06569 D0M6RM 7365 Ki = 13.9 nM T06569 D0N1AW 45485270 Ki = 1300 nM T06569 D0NN3Q 78105 Ki = 1275 nM T06569 D0OI1H 72894 Ki = 772 nM T06569 D0OT5L 1631814 Ki = 7400 nM T06569 D0P6AM 3526523 Ki = 4680 nM T06569 D0Q7DJ 10742 Ki = 7550 nM T06569 D0R4WJ 16129778 Ki = 17800 nM T06569 D0R7QY 127676 Ki = 1860 nM T06569 D0RB0D 44268050 Ki > 500000 nM T06569 D0TY8X 31036 Ki = 86 nM T06569 D0U4BB 10748 Ki = 5500 nM T06569 D0V9EN 689043 Ki = 7330 nM T06569 D0VD7H 84724 Ki = 798 nM T06569 D0X5HL 15107 Ki = 640 nM T06569 D0X6IE 4422372 Ki = 55 nM T06569 D0Y3TZ 370 Ki = 6130 nM T06569 D0YU8J 1502014 Ki = 1097 nM T06569 D0Z1HY 67136 Ki = 608 nM T06569 D0ZC3W 6269 Ki = 1582 nM T03529 D07XOD 2733079 IC50 = 11000 nM T03529 CCI13U 11536910 IC50 = 20400 nM T03529 CN8LG9 13171484 IC50 = 37000 nM T03529 CXC3W5 20377108 IC50 = 28400 nM T03529 C3PDB6 20377110 IC50 = 122000 nM T03529 CI3Q2W 25125116 IC50 = 312000 nM T03529 C5NER0 25125122 IC50 = 7100 nM T03529 CGF7A0 25125458 IC50 = 12800 nM T03529 CS1RD3 25125461 IC50 = 7600 nM T03529 CJ4I7C 25125799 IC50 = 31600 nM T03529 CM6EV5 70681820 IC50 = 7500 nM T03529 CUYZ39 70681821 IC50 = 5600 nM T03529 C9BP5R 70681822 IC50 = 5200 nM T03529 CP6E4R 70681828 IC50 = 16400 nM T03529 CBHO57 70681829 IC50 = 11800 nM T03529 COQC31 70681830 IC50 = 17500 nM T03529 CUF80Q 70681831 IC50 = 15700 nM T03529 CXU67P 70681832 IC50 = 119000 nM T03529 C45NUH 70681833 IC50 = 70600 nM T03529 CV91MS 70681834 IC50 = 194000 nM T03529 CDN0C4 70683924 IC50 = 39800 nM T03529 CH2PL3 70683932 IC50 = 9900 nM T03529 C8E4JH 70683933 IC50 = 7700 nM T03529 CA27DC 70683934 IC50 = 98000 nM T03529 CUC9K6 70686055 IC50 = 17200 nM T03529 C48CLJ 70686056 IC50 = 12300 nM T03529 C59QXF 70688191 IC50 = 21300 nM T03529 C3S9IJ 70688192 IC50 = 11600 nM T03529 C1S3IH 70690203 IC50 = 11400 nM T03529 CJ5PK6 70690208 IC50 = 56000 nM T03529 CL0JW1 70692374 IC50 = 16200 nM T03529 CNW8O1 70692382 IC50 = 13200 nM T03529 CM2KW1 70692383 IC50 = 8400 nM T03529 C04XZL 70694433 IC50 = 6200 nM T03529 CD5O8R 70694437 IC50 = 9500 nM T03529 CTLH58 70696507 IC50 = 10900 nM T03529 C3TV8N 70696508 IC50 = 18700 nM T03529 D05AMQ 6539137 IC50 = 83500 nM T03529 D0M5DR 57330144 IC50 = 36100 nM T97822 D03RTS 2662 IC50 = 89 nM T97822 D0GY5Z 2244 IC50 = 15000 nM T97822 D0R1RS 3715 IC50 = 10 nM T97822 D0U2FN 71321 IC50 = 6500000 nM T97822 D05WPQ 6438354 IC50 = 3200 nM T97822 D09QRO 55390 IC50 = 10000 nM T97822 D0DP8P 47795 IC50 = 5800 nM T97822 D0JY4Y 443292 IC50 > 100000 nM T97822 D0N1SU 133021 IC50 = 160 nM T97822 D0O8ZE 5059 IC50 = 5300 nM T97822 D0S8YL 3969 IC50 = 44000 nM T97822 CH0L7P 71697 IC50 = 950000 nM T97822 CI5D9O 92656 IC50 = 100 nM T97822 CV7L0G 112230 IC50 = 100000000 nM T97822 CT2XZ0 116545 IC50 = 7079457.84 nM T97822 CAT4E3 129615 IC50 = 3388441.56 nM T97822 CCJ76H 512829 IC50 = 9000 nM T97822 CE2BC3 512830 IC50 = 14000 nM T97822 C16VBD 512831 IC50 = 12000 nM T97822 CT7E6Y 573683 IC50 > 800000 nM T97822 CZ0AH3 638278 IC50 = 130000 nM T97822 C6EVL8 854057 IC50 = 3467368.5 nM T97822 CQM64G 3037018 IC50 = 800 nM T97822 COH1C4 3052566 IC50 = 446683.59 nM T97822 C82IPJ 3052567 IC50 = 912010.84 nM T97822 C4VBK3 3253091 IC50 = 50000 nM T97822 CU86JL 4618600 IC50 = 40000 nM T97822 C4M1JC 5709318 IC50 = 44000 nM T97822 COQ7T3 5973690 IC50 = 63000 nM T97822 C3G7DT 6365297 IC50 = 4200 nM T97822 C40FZG 6366698 IC50 = 1300 nM T97822 C02AQY 6366699 IC50 ~ 1000 nM T97822 CWK1F9 6438990 IC50 = 110 nM T97822 C62UOZ 6439221 IC50 = 780 nM T97822 CHQ4Z3 6439222 IC50 = 1300 nM T97822 COC86Q 6439421 IC50 = 390 nM T97822 CLJ91K 6439912 IC50 = 260 nM T97822 C82TEX 7515046 IC50 < 10000 nM T97822 CUS6L8 9822795 IC50 = 30 nM T97822 C5C9ET 10042219 IC50 > 100000 nM T97822 C9T7YV 10063338 IC50 > 100000 nM T97822 CBL7R3 10220019 IC50 = 400 nM T97822 C2WE0I 10246235 IC50 = 9600 nM T97822 C20BTQ 10313997 IC50 = 5500 nM T97822 C8EQI3 10334136 IC50 > 100000 nM T97822 CC1UF0 10335738 IC50 > 100000 nM T97822 C25MYB 10425738 IC50 > 100000 nM T97822 CPR7J0 10469807 IC50 = 12589254.12 nM T97822 C6JI5F 10492615 IC50 > 300000 nM T97822 C0NRO9 10513373 IC50 = 570000 nM T97822 CK0OL2 10704667 IC50 = 27000 nM T97822 CUOI16 10729548 IC50 = 26000 nM T97822 C8IBM2 10801359 IC50 = 250000 nM T97822 CC8S6O 10801786 IC50 = 37000 nM T97822 CDZ94R 10826230 IC50 = 29000 nM T97822 CGLQ72 11723348 IC50 > 100000 nM T97822 CH9VC8 13245625 IC50 > 10000 nM T97822 CRA87I 13556944 IC50 = 14125375.45 nM T97822 C0P5AK 13914227 IC50 > 100000 nM T97822 C49OGE 13914253 IC50 > 100000 nM T97822 C4U3RD 14006855 IC50 = 5000 nM T97822 C6EZ0K 14312565 IC50 > 10000 nM T97822 C2X8PQ 14416570 IC50 = 34 nM T97822 C5PT1G 14416572 IC50 670 nM T97822 C1SG0F 14416576 IC50 = 10000 nM T97822 CRYI80 14416580 IC50 = 610 nM T97822 C27NOS 14416585 IC50 < 10000 nM T97822 C6BP2F 14416587 IC50 < 1000 nM T97822 CER87K 14762923 IC50 = 13803842.65 nM T97822 CGYF09 14762938 IC50 = 501187233.6 nM T97822 CX9AH8 14762939 IC50 = 501187233.6 nM T97822 CU3OT4 14762940 IC50 = 165958690.7 nM T97822 CXT3B5 14762942 IC50 = 100000000 nM T97822 CNZ45J 14762943 IC50 = 91201083.94 nM T97822 CL2A1E 14762944 IC50 = 91201083.94 nM T97822 C78IHC 14762948 IC50 = 50118723.36 nM T97822 CBL2O8 14762951 IC50 = 14791083.88 nM T97822 C8NKZ7 14762954 IC50 = 7079457.84 nM T97822 C4PS0F 14771889 IC50 < 10000 nM T97822 CV41BE 14771890 IC50 = 3100 nM T97822 CCX7K5 14771891 IC50 = 1400 nM T97822 CG57JP 14771892 IC50 = 1300 nM T97822 C91VJM 14771893 IC50 = 230 nM T97822 C0EMA5 14771894 IC50 < 1000 nM T97822 CZ4WJ2 14771895 IC50 = 730 nM T97822 CV5YH8 14771896 IC50 < 10000 nM T97822 C3HNQ2 14771897 IC50 < 10000 nM T97822 CH0TC9 14771898 IC50 < 10000 nM T97822 CX3N7Z 14771899 IC50 = 11000 nM T97822 CX7VA0 14771900 IC50 < 10000 nM T97822 CZC2D4 14771901 IC50 < 10000 nM T97822 CTY60Q 14771902 IC50 < 10000 nM T97822 C0D5OC 14771903 IC50 = 1500 nM T97822 CS3V5C 14771904 IC50 < 10000 nM T97822 CNH5M1 14771905 IC50 = 3200 nM T97822 CXN94C 14771906 IC50 = 510 nM T97822 CY2HF8 14771907 IC50 = 1400 nM T97822 CP5M9A 14771908 IC50 = 190 nM T97822 CI3XK7 14771909 IC50 < 10000 nM T97822 C8NTK2 14771910 IC50 = 750 nM T97822 C8H6XA 14771911 IC50 = 2500 nM T97822 CK53TR 14771912 IC50 < 1000 nM T97822 C10DIY 14771913 IC50 < 1000 nM T97822 C2F9TX 14771915 IC50 = 1100 nM T97822 C83VPQ 14771916 IC50 = 710 nM T97822 CA0C7U 14771917 IC50 = 1000 nM T97822 CK0AR5 14771918 IC50 < 1000 nM T97822 C8SRH6 14771919 IC50 > 10000 nM T97822 CCS9Y4 14771920 IC50 > 10000 nM T97822 C47LJK 14771921 IC50 > 10000 nM T97822 C9OWP0 14771922 IC50 = 1300 nM T97822 C1Z6FX 14771923 IC50 = 780 nM T97822 CHI8M3 14771924 IC50 < 10000 nM T97822 C4JX5S 14771927 IC50 = 590 nM T97822 CRGJ45 14771928 IC50 < 10000 nM T97822 C7L2ZJ 14771929 IC50 = 400 nM T97822 CXAG49 14771930 IC50 < 1000 nM T97822 C54ITL 14771931 IC50 = 110 nM T97822 CC4LM1 14771932 IC50 < 10000 nM T97822 CU6TO3 14771933 IC50 < 10000 nM T97822 C08CRZ 14771934 IC50 = 630 nM T97822 CA3D5U 14771935 IC50 = 1000 nM T97822 CZU2H5 14771936 IC50 = 300 nM T97822 C3B0LX 14771937 IC50 < 10000 nM T97822 CRT9E4 14771938 IC50 > 10000 nM T97822 C18DXV 14977360 IC50 = 71000 nM T97822 CD8YK4 15256755 IC50 = 140000 nM T97822 C53TQI 19044744 IC50 > 100000 nM T97822 CGPW68 19044748 IC50 > 100000 nM T97822 CLN6S5 19044753 IC50 > 100000 nM T97822 CR1W2E 19934882 IC50 > 100000 nM T97822 CF30ID 23275601 IC50 = 66069344.8 nM T97822 CUC36F 23680215 IC50 = 9772372.21 nM T97822 CN6F4H 23680216 IC50 = 4365158.32 nM T97822 C2JUV4 23680221 IC50 = 17782794.1 nM T97822 CHY73S 23680224 IC50 = 524807460.3 nM T97822 C7HV8Y 23680227 IC50 = 70794578.44 nM T97822 CZV8U1 23680228 IC50 = 4677351.41 nM T97822 C54NWH 23680229 IC50 = 741310241.3 nM T97822 CNU43B 23680230 IC50 = 891250938.1 nM T97822 C8A9UV 23689693 IC50 = 562341325.2 nM T97822 CJ1Z9S 44315480 IC50 = 794328234.7 nM T97822 C7UG4F 44315519 IC50 = 15135612.48 nM T97822 C8FEV0 44319113 IC50 = 25000 nM T97822 C1ZH6U 90664380 IC50 > 100000 nM T97822 C5T4EQ 131801158 IC50 = 23 nM T97822 C6JF0E 135616214 IC50 = 2500 nM T97822 CH4YE6 135987613 IC50 > 10000 nM T97822 CFNO28 145950339 IC50 = 34 nM T97822 CG37FR 145950583 IC50 = 27 nM T97822 CCN16Y 145952805 IC50 = 44 nM T97822 C2FVO7 145953074 IC50 = 38 nM T97822 C19TPY 145958203 IC50 = 50 nM T97822 C1BLR8 145959460 IC50 = 33 nM T97822 CUXQ13 145971245 IC50 = 41 nM T97822 C8U9TX 145971276 IC50 = 28 nM T97822 D00GBX 71751 IC50 = 5.7 nM T97822 D01TOR 667555 IC50 = 50000 nM T97822 D05EMX 14076674 IC50 = 10000000 nM T97822 D06VWH 11758240 IC50 = 2 nM T97822 D08GOT 13752584 IC50 = 4897788.19 nM T97822 D09AUL 10266864 IC50 = 51000 nM T97822 D0EW3L 5281222 IC50 = 120000 nM T97822 D0M6UM 129265 IC50 = 22000 nM T97822 D0P1LP 7090 IC50 = 12000 nM T97822 D0U0YE 14762941 IC50 = 165958690.7 nM T97822 D0U2YL 131820 IC50 = 36000 nM T97822 D0U8YQ 921562 IC50 = 14000 nM T23673 D00STL 644241 IC50 = 1100 nM T23673 D05ROI 44462760 IC50 = 150 nM T23673 D09GDD 11167602 IC50 = 1.5 nM T23673 D0E6XR 3062316 IC50 = 164 nM T23673 D0R0MW 5329102 IC50 > 10000 nM T23673 D0W5HK 216239 IC50 = 3 nM T23673 D0Y9EW 42611257 IC50 = 48 nM T23673 D03AND 11656518 IC50 = 19 nM T23673 D04AHQ 71721540 IC50 = 42 nM T23673 D0B9BU 6918454 IC50 = 12 nM T23673 D0E3TC 44259 IC50 = 130 nM T23673 D0F5JZ 24180719 Ki = 3.3 nM T23673 D0M6BD 16719221 IC50 = 56 nM T23673 D0N8RV 9868037 IC50 = 41 nM T23673 D0T4QA 90456533 IC50 = 0.2 nM T23673 D03BNU 59604787 IC50 > 3500 nM T23673 D02YAQ 6603857 IC50 = 49000 nM T23673 D0A9KI 9863367 IC50 > 50 nM T23673 D0F8DL 176155 IC50 = 330 nM T23673 D0T3ME 156422 IC50 = 1400 nM T23673 CB37VR 5034 IC50 = 77 nM T23673 C1YNB7 447721 IC50 > 1000 nM T23673 C73DGZ 656907 IC50 > 1000 nM T23673 CXJ40G 667570 IC50 = 1300 nM T23673 C3OKI4 1228884 IC50 = 1300 nM T23673 C1SVD2 2132479 IC50 = 6500 nM T23673 CVE5C7 2807754 IC50 = 6800 nM T23673 CK2QF5 4163701 IC50 = 17000 nM T23673 C2N9KR 5353919 IC50 = 9 nM T23673 C3G5DZ 9797863 IC50 = 6700 nM T23673 C1A0GW 9798540 IC50 = 1100 nM T23673 CR6T9K 9800910 IC50 = 11000 nM T23673 CNJE78 9811391 IC50 = 1500 nM T23673 CJ7TP1 9818992 IC50 = 4000 nM T23673 C5TVQ1 9819877 IC50 = 230 nM T23673 C1F0PU 9819906 IC50 = 3100 nM T23673 CY52NF 9819987 IC50 = 1200 nM T23673 C8Y9EF 9820630 IC50 = 2000 nM T23673 C1E2DV 9826083 IC50 > 10000 nM T23673 CSQ85J 9827373 IC50 = 700 nM T23673 CP1KY2 9827920 IC50 = 100 nM T23673 C36KUT 9842995 IC50 = 6000 nM T23673 C8UY4X 9844334 IC50 = 6600 nM T23673 C65RQN 9849174 IC50 = 6 nM T23673 C41QWA 9857146 IC50 = 5800 nM T23673 C1W4JG 9872939 IC50 = 400 nM T23673 C45ENX 9883939 IC50 = 3000 nM T23673 CVW95E 9884589 IC50 = 4900 nM T23673 C9KO2G 9884742 IC50 = 7600 nM T23673 CSZ72R 9884877 IC50 = 3700 nM T23673 C18HKQ 9885748 IC50 = 24000 nM T23673 CJ4QV2 9885993 IC50 = 470 nM T23673 CXTE43 9905562 IC50 = 3000 nM T23673 CG47NJ 9906915 IC50 = 6000 nM T23673 C5GE7T 9917045 IC50 = 880 nM T23673 C24UQF 9927821 IC50 = 11000 nM T23673 C5NE6S 9928371 IC50 = 8000 nM T23673 CJT0A3 9929998 IC50 = 7700 nM T23673 C3V6WA 9930407 IC50 = 500 nM T23673 CQ64LI 9935852 IC50 = 695 nM T23673 C61KBJ 9943464 IC50 = 7200 nM T23673 C5ZVD1 9949990 IC50 = 5000 nM T23673 C60EDC 9950128 IC50 = 1700 nM T23673 CW2N9R 9950282 IC50 = 590 nM T23673 CI4BL2 9950385 IC50 = 120 nM T23673 C30RGW 9950906 IC50 = 11000 nM T23673 C3MSR9 9950907 IC50 = 8100 nM T23673 C48ITV 9951822 IC50 = 1900 nM T23673 C2W3AV 9995236 IC50 > 100000 nM T23673 C26QHZ 10005638 IC50 > 10000 nM T23673 CBL7Y0 10127660 IC50 = 53 nM T23673 C0SB5R 10128380 IC50 = 88 nM T23673 CO2E8Y 10128955 IC50 = 73 nM T23673 C30ULG 10128960 IC50 = 410 nM T23673 CABY28 10129238 IC50 = 160 nM T23673 C4V8FQ 10151557 IC50 = 13 nM T23673 C9ZN8M 10151709 IC50 = 61 nM T23673 CS89XI 10152022 IC50 = 300 nM T23673 CLY75M 10173949 IC50 = 130 nM T23673 C6MYH8 10175138 IC50 = 160 nM T23673 C50CXW 10195382 IC50 = 50 nM T23673 C25XBS 10195523 IC50 = 330 nM T23673 C52OSM 10195599 IC50 = 26 nM T23673 C6T3MD 10196590 IC50 = 70 nM T23673 C5E7HJ 10217017 IC50 = 1 nM T23673 C1E6OC 10217682 IC50 = 2300 nM T23673 CE31PD 10218746 IC50 = 210 nM T23673 CLV62C 10238782 IC50 = 460 nM T23673 C2TO8Y 10239830 IC50 = 82 nM T23673 C5WCZ2 10269141 IC50 = 20000 nM T23673 CKF79I 10289214 IC50 = 110 nM T23673 CY6UR3 10289414 IC50 = 100 nM T23673 C26OJV 10289677 IC50 = 150 nM T23673 C3I0MT 10289813 IC50 = 230 nM T23673 CMF93A 10293379 IC50 = 12000 nM T23673 C59HOA 10310634 IC50 = 130 nM T23673 CIO14B 10311595 IC50 = 27 nM T23673 CSAJ01 10311596 IC50 = 170 nM T23673 CZKA14 10311642 IC50 = 44 nM T23673 CSR83F 10311959 IC50 = 63 nM T23673 C17NJQ 10312001 IC50 = 140 nM T23673 CRIA28 10312314 IC50 = 60 nM T23673 CIS0N3 10323382 IC50 = 3500 nM T23673 CA8B5T 10390073 IC50 = 2100 nM T23673 CD47LT 10522840 IC50 = 2600 nM T23673 CN2TU0 10526792 IC50 = 1000 nM T23673 C9Q5ON 10546780 IC50 = 1400 nM T23673 CXN40D 10565927 IC50 = 380 nM T23673 CGSD37 10567785 IC50 = 135 nM T23673 C8E3NI 10568528 IC50 = 90 nM T23673 CFP95Y 10591281 IC50 = 750 nM T23673 CW1L8E 10591928 IC50 = 110 nM T23673 C2JVA6 10595034 IC50 = 20 nM T23673 CJ2O7T 10601190 IC50 = 4500 nM T23673 C16KBG 10637813 IC50 = 5000 nM T23673 C0QC5K 10638921 IC50 = 23 nM T23673 C46ERK 10639924 IC50 = 210 nM T23673 CLSA43 10663963 IC50 = 2100 nM T23673 CTA89W 10664281 IC50 = 610 nM T23673 CK4EW1 10664282 IC50 = 56 nM T23673 CD94OB 10665884 IC50 = 320 nM T23673 CWM72U 10666557 IC50 = 1600 nM T23673 C2UFM7 10711296 IC50 = 950 nM T23673 C1FZ3L 10757716 IC50 = 3000 nM T23673 C29ITE 10829679 IC50 = 86 nM T23673 CKZ95C 10829684 IC50 = 80 nM T23673 C81JVA 10833164 IC50 = 2500 nM T23673 CP6K0I 11155829 IC50 = 210 nM T23673 CSK2W9 11166166 IC50 = 580 nM T23673 CXC91Z 11167118 IC50 = 76 nM T23673 CT1K6D 11167921 IC50 = 180 nM T23673 CZKL03 11190042 IC50 = 120 nM T23673 CGS76Q 11224163 IC50 = 200 nM T23673 C2W5RC 11235063 IC50 > 30000 nM T23673 C6QLP2 11235672 IC50 = 110 nM T23673 C8YQ6T 11235899 IC50 = 170 nM T23673 CH73GV 11258258 IC50 = 480 nM T23673 C2XQC6 11259227 IC50 = 280 nM T23673 CJ69GI 11283035 IC50 = 80 nM T23673 CC1K4L 11294093 IC50 = 490 nM T23673 CQ8CM9 11305234 IC50 = 140 nM T23673 C72GHB 11318236 IC50 = 230 nM T23673 CNFT61 11364677 IC50 = 340 nM T23673 CD57AN 11373388 IC50 = 190 nM T23673 CV24KW 11407374 IC50 = 360 nM T23673 C8W5UG 11407870 IC50 = 250 nM T23673 CFHN02 11407902 IC50 = 340 nM T23673 COT0F6 11418292 IC50 = 480 nM T23673 CP0WH6 11419121 IC50 = 240 nM T23673 C0APW4 11422034 IC50 = 1200 nM T23673 CM3ZU2 11429946 IC50 = 320 nM T23673 CIQ9K8 11430708 IC50 = 550 nM T23673 CD2R4S 11430860 IC50 = 160 nM T23673 C8DA5W 11454055 IC50 = 250 nM T23673 CX7ZP1 11454895 IC50 = 450 nM T23673 CEKC20 11477628 IC50 = 230 nM T23673 CVT10K 11487778 IC50 = 810 nM T23673 CB6ME8 11503895 IC50 = 9 nM T23673 CRP2U5 11526671 Ki > 50000 nM T23673 CO9KP5 11583459 IC50 > 10000 nM T23673 C4U7HM 11621097 IC50 = 116 nM T23673 CU0E8O 11690457 Ki > 10000 nM T23673 C8JW5Z 11696578 IC50 = 38150 nM T23673 CB0AP2 11705863 Ki > 10000 nM T23673 CGI1D9 11717001 Ki = 0.54 nM T23673 CZY05V 11719421 IC50 = 68 nM T23673 C63CKJ 11750387 IC50 = 370 nM T23673 CH3JL9 11750681 IC50 = 190 nM T23673 CO09LN 11750815 IC50 = 260 nM T23673 C8L9ZM 11751978 IC50 = 200 nM T23673 CT8P5W 11775428 IC50 = 660 nM T23673 CIY7C5 12972078 IC50 = 18 nM T23673 C89WYZ 16038368 IC50 > 10000 nM T23673 CZK8V6 16043304 IC50 > 10000 nM T23673 C9TU1O 16046126 IC50 > 1000 nM T23673 C2FR4D 16049771 IC50 = 4 nM T23673 CKV4G1 16079040 IC50 = 1600 nM T23673 C2IF3P 16678352 IC50 = 180 nM T23673 C3IO1C 16679060 IC50 = 1700 nM T23673 C0H8UN 16730109 IC50 > 30000 nM T23673 C8G9AL 16756850 IC50 > 10000 nM T23673 C8M6LZ 17755310 IC50 = 19 nM T23673 CE14ZT 17941505 IC50 = 800 nM T23673 CAF63H 18322354 IC50 = 13000 nM T23673 C14YFA 21024387 IC50 = 170 nM T23673 C4AK5J 21037180 IC50 = 4 nM T23673 C9YR7W 21037208 IC50 = 18 nM T23673 C8ID6R 21037243 IC50 = 41 nM T23673 C2V1EQ 21037245 IC50 = 2 nM T23673 C9MTS8 21037247 IC50 = 9 nM T23673 C1TBC5 21037266 IC50 = 4 nM T23673 CZ23BW 21037364 IC50 = 9 nM T23673 C1CA7H 22040368 IC50 = 53 nM T23673 CG67FQ 22040397 IC50 = 12 nM T23673 CJ4E1M 22040403 IC50 = 780 nM T23673 CSJ67N 22040407 IC50 = 1 nM T23673 C8VJ3A 22040410 IC50 = 210 nM T23673 CHFO54 22040436 IC50 = 1 nM T23673 C19FQT 22040598 IC50 = 1 nM T23673 CJ3UH0 22040625 IC50 = 4 nM T23673 C02DQZ 22040627 IC50 = 20 nM T23673 CCA1D7 22040647 IC50 = 19 nM T23673 C4RP8N 22040656 IC50 = 15 nM T23673 CFK41E 22040722 IC50 = 120 nM T23673 C9A4LW 22040760 IC50 = 14 nM T23673 CSKZ32 22040783 IC50 = 150 nM T23673 CLX26F 22040796 IC50 = 110 nM T23673 CI3V6C 22040802 IC50 = 48 nM T23673 C9WU0J 22040805 IC50 = 490 nM T23673 CDN61H 22040847 IC50 = 10 nM T23673 C3SX8H 22040857 IC50 = 950 nM T23673 CJCL02 22040865 IC50 = 4 nM T23673 C6NM3T 22040925 IC50 = 28 nM T23673 CC84UT 22040937 IC50 = 150 nM T23673 CZM5W1 22040941 IC50 = 6 nM T23673 C30PJQ 22040960 IC50 = 7 nM T23673 CNI32B 22040966 IC50 = 2 nM T23673 C6FMB5 22040978 IC50 = 45 nM T23673 C9A1HQ 22041020 IC50 = 200 nM T23673 CKT6M2 22041042 IC50 = 7300 nM T23673 CM50PH 22041067 IC50 = 27 nM T23673 CRJ4H3 22041111 IC50 = 3500 nM T23673 CO37NP 22041112 IC50 = 1100 nM T23673 C4UMZ2 22041119 IC50 = 56 nM T23673 CI5KM3 22041171 IC50 = 9 nM T23673 C51FDU 22041175 IC50 = 8 nM T23673 CR3G0K 22041260 IC50 = 3 nM T23673 C69BSO 22041261 IC50 = 15 nM T23673 CU85MA 22041278 IC50 = 2 nM T23673 CGX61W 22041319 IC50 = 4 nM T23673 C7HUS0 23585267 IC50 = 28 nM T23673 CHQ23N 23585318 IC50 = 16 nM T23673 COSI68 23585320 IC50 = 11 nM T23673 CV9U8E 24745781 IC50 > 10000 nM T23673 C6JCE7 24753323 IC50 = 26 nM T23673 C50GZI 24753409 IC50 = 13 nM T23673 CC4RZ6 24753410 IC50 = 530 nM T23673 CB3D1Y 24753411 IC50 = 180 nM T23673 C6JF2R 24753412 IC50 = 5 nM T23673 CWX89I 24753603 IC50 = 220 nM T23673 C4CY3V 24753607 IC50 = 300 nM T23673 CQJ2D3 24753784 IC50 = 8 nM T23673 CP1E4R 24753786 IC50 = 32 nM T23673 CA3I4T 24753787 IC50 = 8 nM T23673 CW36DL 24753877 IC50 = 120 nM T23673 COAY09 24753878 IC50 = 23 nM T23673 C9H7EZ 24753971 IC50 = 1500 nM T23673 C6CT7I 24753973 IC50 = 63 nM T23673 CS98MR 24754053 IC50 = 6 nM T23673 C9Q3DE 24754054 IC50 = 4 nM T23673 CRJ9G6 24754132 IC50 = 4 nM T23673 CBD59Z 24754133 IC50 = 45 nM T23673 CKV76A 24754134 IC50 = 37 nM T23673 CM8HY9 24754207 IC50 = 3600 nM T23673 C7YG1N 24759534 IC50 = 630 nM T23673 CCS1U0 24862785 IC50 = 6 nM T23673 C6R4ZU 24863189 IC50 = 1520 nM T23673 CUIS63 24878671 IC50 = 6960 nM T23673 CBUG02 24879141 IC50 > 100000 nM T23673 C2F6KO 24879328 IC50 = 20260 nM T23673 C43HWQ 24883287 IC50 = 10000 nM T23673 C8DA5Q 24883334 IC50 = 10000 nM T23673 C13QYB 24884503 IC50 = 25 nM T23673 C5E1YD 24891645 IC50 = 5840 nM T23673 CY8L7E 24896769 IC50 > 10000 nM T23673 CJZE02 24963588 IC50 = 27 nM T23673 C3DI7Y 24995523 IC50 = 100 nM T23673 CS3Q8B 24995659 IC50 > 2000 nM T23673 CUJZ08 25059320 IC50 = 3200 nM T23673 C2ICS7 25065806 IC50 = 21 nM T23673 CA61PS 25066845 IC50 = 14 nM T23673 CR46MG 25066846 IC50 = 1 nM T23673 CF5AO8 25093353 IC50 > 10000 nM T23673 CAB5K2 25114576 IC50 = 870 nM T23673 C9PL5S 25137959 IC50 = 2000 nM T23673 CVJ0S5 25137960 IC50 = 10 nM T23673 C6FGQ1 25206346 IC50 = 23 nM T23673 CC71QJ 27666048 IC50 > 100000 nM T23673 CIJ56L 44142782 IC50 > 10000 nM T23673 CCFQ29 44187005 IC50 = 8.52 nM T23673 CR7K2T 44223999 Ki = 0.3 nM T23673 CJ75IB 44250343 IC50 = 120 nM T23673 CS2CK9 44250550 IC50 = 105 nM T23673 CLY1A3 44251218 IC50 = 200 nM T23673 C4O0CH 44272164 IC50 = 18000 nM T23673 CX28HG 44272165 IC50 = 18000 nM T23673 CNIJ29 44309757 IC50 > 10000 nM T23673 CH1TA5 44309758 IC50 = 570 nM T23673 C4P9ZA 44312235 IC50 = 29 nM T23673 CX57BA 44312236 IC50 = 40 nM T23673 C2D7RK 44312254 IC50 = 32 nM T23673 C8MF2U 44312272 IC50 = 65 nM T23673 C4XCW8 44312367 IC50 = 25 nM T23673 CGRP10 44312380 IC50 = 16 nM T23673 C2IC8R 44326529 IC50 = 15000 nM T23673 CT74PB 44326530 IC50 = 12000 nM T23673 C1W6BM 44326737 IC50 = 25000 nM T23673 CO0UF5 44326798 IC50 = 19000 nM T23673 C0E4TU 44326810 IC50 = 16000 nM T23673 C0GRN1 44326814 IC50 = 15000 nM T23673 CV37KZ 44326926 IC50 = 22000 nM T23673 C4ZD0E 44326936 IC50 = 20000 nM T23673 C0KD4U 44346053 IC50 = 8700 nM T23673 CO0FN8 44378490 IC50 = 130 nM T23673 CR1MV0 44378504 IC50 = 68 nM T23673 C4D5ZM 44378534 IC50 = 120 nM T23673 CI3W6L 44378535 IC50 = 38 nM T23673 C39PLZ 44378637 IC50 = 500 nM T23673 C9E7ID 44378798 IC50 = 270 nM T23673 C7HGZ5 44378800 IC50 = 460 nM T23673 CBGZ52 44378801 IC50 = 140 nM T23673 CIV90F 44378900 IC50 = 130 nM T23673 CI6T9Z 44378901 IC50 = 5800 nM T23673 C6CW1H 44378902 IC50 = 370 nM T23673 CJH86A 44385063 IC50 > 50000 nM T23673 CG46BQ 44386338 IC50 > 10000 nM T23673 CJTF35 44418481 IC50 = 100 nM T23673 CKV61A 44418488 IC50 = 630 nM T23673 CJ49OD 44418525 IC50 = 1000 nM T23673 C8LB9S 44418539 IC50 = 250 nM T23673 CO8X1V 44418540 IC50 = 158 nM T23673 C1IX6V 44418547 IC50 = 251 nM T23673 C4Q5UL 44418563 IC50 = 40 nM T23673 C8NZ9D 44418572 IC50 = 10 nM T23673 CJ3DL4 44418573 IC50 = 7 nM T23673 C10MKH 44448311 IC50 = 49 nM T23673 C1QN4V 44448333 IC50 = 41 nM T23673 CLQF97 44448334 IC50 = 26 nM T23673 C73THQ 44448354 IC50 = 5 nM T23673 C0DPU3 44448725 IC50 = 2 nM T23673 CFQN07 44448726 IC50 = 17 nM T23673 CR85LO 44448746 IC50 = 20 nM T23673 C5Y2JR 44448747 IC50 = 1 nM T23673 CA76JX 44448748 IC50 = 0.5 nM T23673 C9I0DU 44453753 IC50 = 6300 nM T23673 C2T7UV 44454440 IC50 = 8600 nM T23673 C0TN9Z 44454441 IC50 = 6300 nM T23673 C3P2TG 44454464 IC50 = 3500 nM T23673 CDN4M7 44565710 IC50 = 44 nM T23673 CB39SW 44565730 IC50 = 160 nM T23673 C13WTF 44565731 IC50 = 230 nM T23673 CEU40V 44565732 IC50 = 440 nM T23673 C6HEU1 44565743 IC50 = 2700 nM T23673 C5VL3A 44565744 IC50 = 4400 nM T23673 CI5M9V 44565745 IC50 = 500 nM T23673 CCD0E2 44565749 IC50 = 700 nM T23673 C4P7KM 44565750 IC50 = 820 nM T23673 CBZ1H2 44565751 IC50 = 1000 nM T23673 C39TYG 44565752 IC50 = 1100 nM T23673 C8QDY6 44565771 IC50 = 7500 nM T23673 CQAB41 44565772 IC50 = 10000 nM T23673 CUK3E8 44565773 IC50 = 650 nM T23673 CK24HZ 44565794 IC50 = 9500 nM T23673 CG0PL1 44565795 IC50 = 1400 nM T23673 C53FHZ 44565817 IC50 = 1500 nM T23673 C9VXN3 44578709 IC50 = 80 nM T23673 C3Y5AW 44589519 IC50 = 41 nM T23673 C09EWJ 44590206 IC50 = 17 nM T23673 CUA97D 46209401 IC50 = 1.4 nM T23673 C2P9QO 46228508 IC50 = 198 nM T23673 C6E5PY 46228822 IC50 = 126 nM T23673 C3T8AM 46228951 IC50 = 3 nM T23673 C4MKC5 46870033 IC50 = 11 nM T23673 C7LK1C 46945257 IC50 = 765 nM T23673 CHSF07 49806372 IC50 > 1000 nM T23673 C5ME3S 49806721 IC50 > 50000 nM T23673 CS7J8G 50937465 IC50 = 79 nM T23673 C2Q0GE 50990922 IC50 = 3000 nM T23673 C61DVY 50990961 IC50 = 2.2 nM T23673 CV3UP9 50992247 IC50 = 2.5 nM T23673 COVJ29 50994971 IC50 = 169 nM T23673 C5X9OM 51354603 IC50 = 10 nM T23673 C4DSG2 51354885 IC50 = 6.2 nM T23673 CQ85FC 51354886 IC50 = 110 nM T23673 C7MOQ0 51354887 IC50 = 70 nM T23673 C5KVT1 51355181 IC50 = 4.5 nM T23673 CS5F4Z 51355182 IC50 = 780 nM T23673 C4NFL7 51355183 IC50 = 3.3 nM T23673 C4W6PY 51355459 IC50 = 4.6 nM T23673 C95FWU 51355461 IC50 = 45 nM T23673 C4J3RE 51355733 IC50 = 6 nM T23673 CEQN27 52936621 Ki > 2000 nM T23673 CM24LF 52938983 IC50 = 2.87 nM T23673 CFR21J 52939107 IC50 = 22.41 nM T23673 CJQ31I 53239946 IC50 = 11 nM T23673 C7B3DE 53239955 IC50 = 13 nM T23673 C8UZE6 53239978 IC50 = 46 nM T23673 C1SKV3 53249125 IC50 = 1 nM T23673 C4CO1V 53317057 IC50 = 240.3 nM T23673 CE73CS 53323686 IC50 = 8319 nM T23673 CFP84X 53324920 IC50 = 1100 nM T23673 CD4H3S 53354074 Ki > 1000 nM T23673 CM7P3W 53357328 IC50 > 50000 nM T23673 CVG90B 53389651 IC50 > 10000 nM T23673 C89YCL 54580728 IC50 = 3 nM T23673 CA9I0J 54580729 IC50 = 4 nM T23673 C4X6DP 54581730 IC50 = 3 nM T23673 C2KHN1 54581731 IC50 = 1 nM T23673 CQ3U7M 54582720 IC50 = 140 nM T23673 C6ZR1A 54583026 IC50 = 530 nM T23673 CP7U4T 54584640 IC50 = 1 nM T23673 CC7T2A 56674921 IC50 = 170 nM T23673 CT4E8R 56832546 IC50 = 8500 nM T23673 CP58NG 56954518 IC50 = 930 nM T23673 CAK91L 56955954 IC50 = 206 nM T23673 C8LZ5B 56966054 IC50 = 10.6 nM T23673 CCE7J3 56966055 IC50 = 75.9 nM T23673 CP10UK 56966056 IC50 = 87.8 nM T23673 CMS50K 56966057 IC50 = 13.1 nM T23673 CRPT61 56966123 IC50 = 69.2 nM T23673 C6X0EZ 56966125 IC50 = 94.9 nM T23673 CLI12D 56966126 IC50 = 120.3 nM T23673 C9L4IJ 56966199 IC50 = 147.9 nM T23673 CTP30L 56966200 IC50 = 77.7 nM T23673 COA5X2 56966201 IC50 = 35.9 nM T23673 CIBO79 56966202 IC50 = 22.1 nM T23673 C2KDZ7 56966273 IC50 = 16.5 nM T23673 CGJ6F0 56966274 IC50 = 64.8 nM T23673 C48QKV 56966276 IC50 = 46.7 nM T23673 C4G7QD 57343225 IC50 = 73 nM T23673 CU4FW8 57397383 IC50 = 1600 nM T23673 C0BGR6 57399335 IC50 = 3 nM T23673 CZSM95 57412684 IC50 > 10000 nM T23673 CVK0G4 58056356 IC50 > 50000 nM T23673 CKB3A4 58102283 IC50 > 10000 nM T23673 CX1G3L 58102286 IC50 = 100 nM T23673 C1R8NM 59139106 IC50 = 78 nM T23673 CB34LP 59139113 IC50 = 120 nM T23673 CWK9I8 59139139 IC50 = 2500 nM T23673 CWN47R 59139154 IC50 = 70 nM T23673 CT0JG1 59139161 IC50 = 16 nM T23673 CP5GY6 59139172 IC50 = 81 nM T23673 CL4X3Z 59139185 IC50 = 70 nM T23673 C1PE3R 59139202 IC50 = 2400 nM T23673 CE82OV 59139228 IC50 = 1100 nM T23673 C3T5OF 59139235 IC50 = 56 nM T23673 CWO17Q 59139262 IC50 = 5 nM T23673 C5IYT0 59139264 IC50 = 25 nM T23673 C91SBH 59139388 IC50 = 830 nM T23673 C62EVK 59139472 IC50 > 50000 nM T23673 CT3EW2 59292007 IC50 > 1000 nM T23673 CXJ63M 59603829 IC50 = 560 nM T23673 CQEU96 59603842 IC50 = 48 nM T23673 C1MR8Q 60097495 IC50 > 10000 nM T23673 C9W0PE 60150671 IC50 = 75 nM T23673 C9NAL6 60152613 IC50 = 0.6 nM T23673 CSZA16 60155724 IC50 = 1814 nM T23673 CW3G6N 60196633 IC50 = 340 nM T23673 CUV14K 60196634 IC50 = 4300 nM T23673 CU32ED 60196737 IC50 = 175 nM T23673 CKB59I 60196738 IC50 > 10000 nM T23673 C40LVZ 60196740 IC50 > 10000 nM T23673 CV63UL 67240318 IC50 > 10000 nM T23673 CW17YX 68281294 IC50 = 1000 nM T23673 C5DGR9 69036886 IC50 = 4012 nM T23673 C4BT3M 69037249 IC50 = 2.9 nM T23673 CVBR46 70696651 IC50 = 81.5 nM T23673 CRX81Q 71575642 IC50 = 72 nM T23673 CT93OP 71682347 IC50 > 10000 nM T23673 C3NV9Q 71682348 IC50 > 10000 nM T23673 CN7M9G 71682349 IC50 = 293 nM T23673 C8KU4O 71682499 IC50 > 10000 nM T23673 C0XEQ1 71682500 IC50 = 30 nM T23673 CXSI14 71718330 IC50 > 100000 nM T23673 C1TM3P 71720141 IC50 > 100000 nM T23673 CU83YL 71730951 IC50 = 2.8 nM T23673 C7F3ZM 71736390 IC50 = 1.6 nM T23673 C9EM5X 71736552 IC50 = 6.7 nM T23673 CKYO24 71736864 IC50 = 5.6 nM T23673 CSVW76 72546488 IC50 = 570 nM T23673 C7HBR1 72546491 IC50 = 40 nM T23673 CXYT34 72546730 IC50 = 56 nM T23673 C1DAW5 72546731 IC50 = 50 nM T23673 C6R8DI 72943374 IC50 = 80 nM T23673 C80SEC 73504974 IC50 = 652 nM T23673 C3KVB2 73505180 IC50 = 92 nM T23673 CP4ZX2 76317169 IC50 = 120 nM T23673 C4DT2Z 76335375 IC50 = 55 nM T23673 CA5O6K 78325057 IC50 = 0.1 nM T23673 CCD78B 86295666 IC50 = 0.2 nM T23673 C2OGP3 86296699 IC50 = 0.2 nM T23673 C80LAH 86298305 EC50 = 200 nM T23673 CI2CG1 89670173 IC50 = 7 nM T23673 C1HW4B 89735655 IC50 = 950 nM T23673 C7TJR3 89814000 IC50 = 1.2 nM T23673 C4WP7D 89827799 IC50 = 7.2 nM T23673 CJE4A5 90407961 IC50 = 0.6 nM T23673 C9KN1H 90408121 EC50 = 52 nM T23673 CF45CE 90408582 IC50 = 0.4 nM T23673 C6RZ7J 90408826 EC50 = 20 nM T23673 CXZ6M2 90408889 EC50 = 76 nM T23673 C7QD9P 90409579 EC50 = 80 nM T23673 CU0GW5 90442604 IC50 = 0.8 nM T23673 CA2E5S 90456597 EC50 = 8 nM T23673 CW6S8P 90655795 IC50 > 50000 nM T23673 CNYK35 90655796 IC50 = 27000 nM T23673 CE4LR9 90655797 IC50 = 21 nM T23673 CWD4O3 90655989 IC50 > 50000 nM T23673 C26BSU 90666124 IC50 = 3200 nM T23673 CVQ1O6 90666126 IC50 = 286 nM T23673 C5AN9J 90666128 IC50 = 4300 nM T23673 CP76NE 90666130 IC50 > 50000 nM T23673 C85GHD 90666131 IC50 = 16500 nM T23673 CRP9I5 90666132 IC50 = 9200 nM T23673 CX1NV3 117609603 EC50 = 3960 nM T23673 CQ40CN 117609669 EC50 = 5 nM T23673 C5XEY9 117610044 EC50 = 64 nM T23673 C8E9JO 117610115 EC50 = 27 nM T23673 CG7QL4 118705925 IC50 = 8.79 nM T23673 C4AHL2 118711367 IC50 > 10000 nM T23673 CQCX41 118737057 IC50 = 27 nM T23673 C9KWP7 118870913 IC50 = 0.4 nM T23673 CSR81B 118887129 EC50 = 21 nM T23673 CV3MY8 118938835 IC50 = 0.1 nM T23673 CU52FB 118938855 IC50 = 0.1 nM T23673 C9NDH0 118938856 IC50 = 2 nM T23673 CTLH73 118938861 IC50 = 0.03 nM T23673 CL4MP3 118938866 IC50 = 6 nM T23673 C0UT7G 122177477 IC50 = 3.1 nM T23673 CSF49R 122177478 IC50 = 5.2 nM T23673 C5B6QT 122189918 IC50 = 44.8 nM T23673 C4X7SD 122192466 IC50 > 10000 nM T23673 CNX0Q2 122193763 IC50 > 10000 nM T23673 CWV0C3 122193764 IC50 = 4020 nM T23673 CSG98Y 122193765 IC50 > 10000 nM T23673 CCLQ75 122193769 IC50 = 6220 nM T23673 CXDR48 122193770 IC50 > 10000 nM T23673 CPA8C5 122193773 IC50 = 5840 nM T23673 CWM37L 123897305 IC50 = 71 nM T23673 CF5WH1 127039888 IC50 = 38600 nM T23673 CAG9K7 127046489 IC50 = 15 nM T23673 C6DP7Y 127047275 IC50 = 111 nM T23673 C3DVM9 127047276 IC50 = 566 nM T23673 CM81AR 127047922 IC50 = 695 nM T23673 CA2C3D 129010136 EC50 = 200 nM T23673 C0FM1R 130196825 IC50 = 27920 nM T23673 CR5P1D 132067922 IC50 = 0.6 nM T23673 CU1H0W 132497402 IC50 = 43.4 nM T23673 CZ81AL 134142029 IC50 = 0.024 nM T23673 C7PS8C 135271570 IC50 = 76 nM T23673 C8B5GZ 135513879 IC50 = 390 nM T23673 CGL3F1 135957036 IC50 = 50 nM T23673 C4REH9 135957052 IC50 = 76 nM T23673 C58FQY 135957053 IC50 = 156 nM T23673 CG9PJ7 135993841 IC50 = 960.9 nM T23673 CUA72Z 136042194 IC50 = 667.8 nM T23673 CL2D1A 136086817 IC50 = 146 nM T23673 CKG0N2 136086821 IC50 = 370 nM T23673 CH70WS 136086832 IC50 = 839 nM T23673 CG1R7B 136087060 IC50 = 6500 nM T23673 CRB3M4 136609929 IC50 = 2500 nM T23673 C0A9VE 136609930 IC50 = 1300 nM T23673 CW5YL0 136609931 IC50 > 50000 nM T23673 C3FC1W 137631894 IC50 = 7500 nM T23673 C7NFX9 137632089 IC50 = 8.5 nM T23673 C0Y1AW 137632207 IC50 = 150 nM T23673 C10BTW 137632556 IC50 > 10000 nM T23673 C2J9GO 137633617 IC50 > 10000 nM T23673 C7MD0H 137635615 IC50 = 28 nM T23673 CML76T 137635976 IC50 = 6200 nM T23673 CS9AW4 137636754 IC50 = 272 nM T23673 C08MHJ 137636777 IC50 = 0.7 nM T23673 CV3A5G 137637973 IC50 = 34.5 nM T23673 C7R0MS 137638615 IC50 = 2300 nM T23673 CE96AL 137639657 IC50 = 17300 nM T23673 CEPU59 137640849 IC50 = 220 nM T23673 CGR5B1 137642299 IC50 = 51 nM T23673 CA13KP 137642491 IC50 = 18.7 nM T23673 C26HIT 137643417 IC50 = 2100 nM T23673 CAT49C 137645403 IC50 = 374 nM T23673 CUES49 137646218 IC50 = 1800 nM T23673 CS6J8X 137646633 IC50 > 10000 nM T23673 C9Z6NB 137646838 IC50 = 770 nM T23673 CL8W4P 137647062 IC50 = 21.4 nM T23673 CGQ02E 137648059 IC50 = 6.3 nM T23673 C2HFR6 137648529 IC50 = 690 nM T23673 CL9HT1 137648599 IC50 = 21.9 nM T23673 CYR2I7 137649411 IC50 = 3050 nM T23673 C17GBS 137649678 IC50 = 1840 nM T23673 CEO70C 137650358 IC50 > 10000 nM T23673 CE7KF3 137650390 IC50 = 13.3 nM T23673 C4NM0R 137650776 IC50 = 1280 nM T23673 C3LAD6 137652990 IC50 > 100000 nM T23673 CL3P8Q 137653011 IC50 = 89 nM T23673 C5B9AM 137653362 IC50 = 860 nM T23673 C8K0OY 137655533 IC50 = 670 nM T23673 C3F8ZD 137656536 EC50 = 700 nM T23673 CMPJ36 137656808 IC50 = 14.4 nM T23673 C83XOY 137657177 IC50 = 53 nM T23673 CF7U5Y 137657487 IC50 > 10000 nM T23673 C3SD7B 137658277 IC50 = 4900 nM T23673 CVY3F0 137658568 IC50 = 1510 nM T23673 CJK81S 137659431 IC50 = 99 nM T23673 CNWY53 137659664 IC50 = 370 nM T23673 CUS48N 137659983 IC50 = 327 nM T23673 CA4V9R 137661906 IC50 = 100 nM T23673 COB9P2 141456067 IC50 = 7900 nM T23673 C6CN8H 142739455 IC50 = 61 nM T23673 CT25FH 145950796 IC50 = 8.5 nM T23673 C2I5WD 145979310 IC50 = 13.3 nM T23673 C6T4MU 145982183 IC50 = 40 nM T23673 CI1VH9 145985185 IC50 > 200000 nM T23673 CI7M2B 145988861 IC50 = 17.5 nM T23673 CNLH48 145988888 IC50 = 17600 nM T23673 CRT48W 145993502 IC50 = 3150 nM T23673 C2NKF8 155076930 IC50 = 182 nM T23673 CY1ZH2 155510358 IC50 = 336 nM T23673 CZ5S2M 155512875 IC50 = 2.7 nM T23673 C2MD1Q 155513187 IC50 > 10000 nM T23673 C0MZ9A 155513534 IC50 = 5160 nM T23673 CI54TD 155514548 IC50 = 1420 nM T23673 C2BA1L 155514841 IC50 = 1310 nM T23673 CX6SR0 155516442 IC50 = 420 nM T23673 CS31UH 155519078 IC50 = 1520 nM T23673 CU6Z5O 155520650 IC50 = 130 nM T23673 CP4JL5 155521754 IC50 = 4490 nM T23673 CVQ35F 155522102 IC50 = 3540 nM T23673 CM3DB7 155523430 IC50 = 480 nM T23673 CLY07C 155530863 IC50 = 450 nM T23673 CVQ24P 155532080 IC50 = 990 nM T23673 CS69CA 155532132 IC50 = 0.5 nM T23673 CJP67I 155535248 IC50 = 5320 nM T23673 C8ZF4H 155544511 IC50 = 3660 nM T23673 C8T0MQ 155544690 IC50 = 840 nM T23673 CJL37G 155544854 IC50 = 16400 nM T23673 CHE5F1 155553390 IC50 = 6260 nM T23673 CYC23K 155560669 IC50 = 110 nM T23673 C81JZW 155563388 IC50 = 410 nM T23673 C62CIM 155565320 IC50 = 420 nM T23673 CH3NO1 155566774 IC50 = 31.7 nM T23673 C0V2MU 135398506 Ki = 1.72 nM T23673 D00NWF 5730 IC50 = 70 nM T23673 D02XHC 448912 IC50 > 100000 nM T23673 D03MUZ 17759555 IC50 > 100000 nM T23673 D05UPS 44418518 IC50 = 398 nM T23673 D06WJA 9950176 IC50 = 1.4 nM T23673 D08LYB 5166 IC50 > 50 nM T23673 D0C0ZC 11676786 IC50 = 380 nM T23673 D0IR6U 5494425 IC50 > 10000 nM T23673 D0J4YA 9943465 IC50 > 12000 nM T23673 D0QN6U 9806182 IC50 = 810 nM T23673 D0V0QJ 389898 IC50 = 34500 nM T23673 D0Z5TQ 5924208 IC50 = 10.6 nM T48598 D05ROI 44462760 IC50 = 5880 nM T48598 D0Y9EW 42611257 IC50 = 16600 nM T48598 D04AHQ 71721540 IC50 = 150 nM T48598 CE2VX1 1381961 IC50 = 155000 nM T48598 C4K3AC 9870962 EC50 = 1065 nM T48598 C3MSB4 9954645 EC50 > 10000 nM T48598 C4BT3M 69037249 IC50 = 91 nM T48598 C3D6WC 71515468 IC50 = 200 nM T48598 CU83YL 71730951 IC50 = 48 nM T48598 C7F3ZM 71736390 IC50 = 46 nM T48598 C9EM5X 71736552 IC50 = 270 nM T48598 CKYO24 71736864 IC50 = 120 nM T48598 C2A4YP 86279165 Ki = 200000 nM T48598 C7TJR3 89814000 IC50 = 16 nM T48598 C4WP7D 89827799 IC50 = 160 nM T48598 CHJ6B8 90665836 IC50 = 1200 nM T48598 CFI02E 90665837 IC50 = 10000 nM T48598 CI6DB8 90665838 IC50 = 1800 nM T48598 C61RVL 90665839 IC50 = 10000 nM T48598 CW2UX9 90665840 IC50 = 10000 nM T48598 CDN49I 90665841 IC50 = 700 nM T48598 C0KI6U 90665842 IC50 = 1100 nM T48598 C0W7UI 90665843 IC50 = 2000 nM T48598 CYU7W2 90665844 IC50 = 2300 nM T48598 CEJ3D4 118019010 IC50 = 496 nM T48598 C0UT7G 122177477 IC50 = 57 nM T48598 CSF49R 122177478 IC50 = 120 nM T48598 CYP1B7 132145599 IC50 > 16000 nM T48598 CG7J5E 132162814 IC50 = 7600 nM T48598 CDWB35 132162815 IC50 > 16000 nM T48598 C1DW2E 132162816 IC50 > 16000 nM T48598 CJ1MY3 132162817 IC50 > 16000 nM T48598 C74FYN 132162819 IC50 > 16000 nM T48598 C2SIJ4 132162853 IC50 = 1900 nM T48598 CB80ZS 132163177 IC50 = 1500 nM T48598 C6CL4S 132163178 IC50 = 540 nM T48598 C3GPQ1 132163222 IC50 = 70 nM T48598 CULE35 135148667 IC50 = 8 nM T48598 C6DYW3 135148885 IC50 = 220 nM T48598 CU8T3N 136346978 Ki = 9 nM T48598 CC20EZ 136346980 Ki = 280 nM T48598 CY2L6T 136346989 Ki = 5000 nM T48598 CUG30Y 136347012 Ki > 25000 nM T48598 CS8YP7 137003167 IC50 = 939 nM T48598 CGS71A 137278705 IC50 = 51 nM T48598 CJ9N2K 137278711 IC50 = 68 nM T48598 C1HX7O 137278713 IC50 = 63 nM T48598 CK4MJ2 137278717 IC50 = 25 nM T48598 CA7GT6 137283289 Ki = 382 nM T48598 CS4W8U 137288869 IC50 = 69 nM T48598 C34DAC 137288870 IC50 = 36 nM T48598 CB42LP 137289789 Ki = 374 nM T48598 C0GNH8 137290307 Ki = 50000 nM T48598 CN2U1R 137290313 Ki = 8000 nM T48598 CX30GO 137290327 Ki = 2200 nM T48598 CW7Y3V 137292511 Ki = 15200 nM T48598 CXM3Y9 137297869 IC50 = 3330 nM T48598 C2XJN7 137297879 IC50 = 903 nM T48598 CRZH30 137297882 IC50 = 101 nM T48598 CBG13S 137297890 IC50 = 1800 nM T48598 C7BL0Z 137297899 IC50 = 7150 nM T48598 C1TWR9 137297909 IC50 = 20100 nM T48598 C85PEX 137297911 IC50 = 28 nM T48598 CS9D7J 137297914 IC50 = 3520 nM T48598 CTU65M 137297915 IC50 = 51 nM T48598 CJY69R 137297923 IC50 = 9150 nM T48598 CTO29V 137303087 Ki > 10000 nM T48598 C9SZ6B 137303128 Ki = 920 nM T48598 CVH3G7 137304434 Ki = 36000 nM T48598 C2LV5C 137304502 Ki = 5000 nM T48598 CV9Q5S 137314428 Ki = 380 nM T48598 CG7F2B 137314429 Ki > 20000 nM T48598 C8KFZ5 137316419 Ki = 2700 nM T48598 CQ7Z4X 137316471 Ki = 1600 nM T48598 C2M5GX 137317563 Ki = 3500 nM T48598 CJ07SA 137636907 IC50 = 50 nM T48598 CFA74W 137637303 IC50 = 64 nM T48598 C17EOK 137637743 IC50 = 1190 nM T48598 C7JU3W 137639238 IC50 = 35.8 nM T48598 CS93CA 137639750 IC50 = 1.6 nM T48598 CUS40W 137643713 IC50 = 59 nM T48598 CN4FM5 137645102 IC50 = 6.1 nM T48598 CK7S3H 137646089 IC50 = 1630 nM T48598 CFT25U 137647500 IC50 = 2.7 nM T48598 CM2XF3 137648559 IC50 = 426 nM T48598 C0UKF3 137648822 IC50 = 764 nM T48598 CP4V6Y 137650846 IC50 = 15400 nM T48598 CRF93P 137650861 IC50 = 19 nM T48598 CXO6C3 137652506 IC50 = 20600 nM T48598 CBIZ98 137653897 IC50 = 243 nM T48598 CLWD10 137660005 IC50 = 83 nM T48598 C78JQW 137661919 IC50 = 11 nM T48598 CKWQ13 138678754 IC50 < 5 nM T48598 CWM42J 138678756 IC50 = 18 nM T48598 C8S1AT 138678759 IC50 = 16 nM T48598 CA18QI 138678764 IC50 = 70 nM T48598 C9J3EN 138678770 IC50 = 132 nM T48598 C6SPK8 138678774 IC50 = 387 nM T48598 C7EV3T 138678780 IC50 = 610 nM T48598 CE7Q0H 138678786 IC50 = 97 nM T48598 C92HTX 138678788 IC50 = 81 nM T48598 C27KFX 138678799 IC50 = 150 nM T48598 C30MEF 138678890 IC50 = 211 nM T48598 C2DOL1 138679046 IC50 = 52 nM T48598 CR5A6H 139388519 IC50 = 780 nM T48598 CYRW58 139388529 IC50 = 4860 nM T48598 C5GLR3 139388566 IC50 = 169 nM T48598 CG1MO4 139388571 IC50 = 116 nM T48598 CNVK52 139388599 IC50 = 129 nM T48598 CXB0Y3 139388605 IC50 = 214 nM T48598 C8CRF6 139600305 IC50 = 115 nM T48598 CEL25S 140956840 IC50 = 11 nM T48598 C0NV4K 140956861 IC50 = 66 nM T48598 C1SJI0 142468965 IC50 = 18 nM T48598 CB29ZR 142468976 IC50 = 12 nM T48598 C9PC5N 142468998 IC50 = 12 nM T48598 C6S0VF 142469011 IC50 = 21 nM T48598 C3PD0Y 142469055 IC50 = 32 nM T48598 C7X6QM 142469058 IC50 = 97 nM T48598 CUW9Y5 146234885 IC50 = 128 nM T48598 CN08TQ 146234893 IC50 = 25 nM T48598 CB30HO 146235053 IC50 = 80 nM T48598 C2B5VH 146235304 IC50 = 47 nM T48598 CKM1C3 146235420 IC50 = 90 nM T48598 C5QBX0 146235429 IC50 = 53 nM T48598 C91ANQ 146235452 IC50 = 142 nM T48598 CAVJ61 146235508 IC50 = 34 nM T48598 CFKC35 146235592 IC50 = 164 nM T48598 C3HCA7 146235786 IC50 = 65 nM T48598 C89YKH 146235843 IC50 = 38 nM T48598 C5KX3F 146235857 IC50 = 306 nM T48598 C42CDB 146235944 IC50 = 53 nM T48598 CQW98L 146236007 IC50 = 146 nM T48598 C76QJC 146236012 IC50 = 56 nM T48598 C06VPI 146254335 IC50 = 109 nM T48598 C0U1KX 146254417 IC50 = 442 nM T48598 CZ7P4M 146254588 IC50 = 25 nM T48598 C3S5WI 146461338 IC50 = 29 nM T48598 CBI9U1 146585881 IC50 = 109 nM T48598 C1EFX9 146585884 IC50 = 683 nM T48598 C3H9BP 146585895 IC50 = 139 nM T48598 C1VJ4L 146630440 IC50 = 17900 nM T48598 C6S1IB 146630461 IC50 = 2120 nM T48598 C9I2WV 146630653 IC50 > 250000 nM T48598 C4IA5T 146630666 IC50 = 299 nM T48598 C51IYS 146630676 IC50 = 638 nM T48598 CW34ZK 146630683 IC50 = 1370 nM T48598 CVL6A5 146630701 IC50 = 4260 nM T48598 C4QH7U 146630731 IC50 = 6630 nM T48598 C0WAB5 146630732 IC50 = 14200 nM T48598 CYH28N 146630894 IC50 = 369 nM T48598 C5IV8H 146630905 IC50 = 1290 nM T48598 CIX1C8 146630907 IC50 = 174 nM T48598 CNK71Q 146631214 IC50 = 1270 nM T48598 C8H9TW 155523678 IC50 = 73 nM T48598 CBR9O0 155524545 IC50 = 4342 nM T48598 CVQ3H7 155528727 IC50 = 7653 nM T48598 C7Y3FZ 155549278 IC50 = 627 nM T48598 CMA86J 155564813 IC50 = 2780 nM T58093 D0S7BQ 52918384 IC50 = 12 nM T58093 D0T2IQ 443600 IC50 = 20 nM T58093 C8A6FD 9849925 IC50 = 30 nM T58093 C04KRJ 16034963 IC50 = 2.5 nM T58093 CJ42NE 16034968 IC50 = 0.52 nM T58093 CEYX96 16035081 IC50 = 0.93 nM T58093 CH97SC 16035085 IC50 = 2.1 nM T58093 CTC5O9 16035087 IC50 = 1.4 nM T58093 C4OQ3K 16035189 IC50 = 1.4 nM T58093 CG83UV 16035293 IC50 = 3.8 nM T58093 CGN4W5 16035295 IC50 = 3.2 nM T58093 CSFC45 16035507 IC50 = 2.2 nM T58093 CNTW74 16035824 IC50 = 12 nM T58093 CCDG98 16035825 IC50 = 5.2 nM T58093 CZC1T5 16035827 IC50 = 8 nM T58093 C48ARB 16036037 IC50 = 4.5 nM T58093 C1SMZ2 16036156 IC50 = 2.2 nM T58093 CP3H6M 16036157 IC50 = 4.4 nM T58093 C9YZ6I 16036158 IC50 = 1.4 nM T58093 C2I1YX 16036160 IC50 = 1.5 nM T58093 C3ZIH1 16036281 IC50 = 2.4 nM T58093 C5SOI2 16036282 IC50 = 3.4 nM T58093 C7JG1B 16036394 IC50 = 10 nM T58093 C3NWE9 16036395 IC50 = 2 nM T58093 CW16UL 16036656 IC50 = 5 nM T58093 C2VOZ5 16036657 IC50 = 4 nM T58093 C3IU1P 16036659 IC50 = 2 nM T58093 C9SHM6 16036661 IC50 = 3.7 nM T58093 CMOB46 16046174 IC50 = 7500 nM T58093 C7WH3R 25123230 IC50 = 30 nM T58093 CV15JQ 25123888 IC50 = 30 nM T58093 CFD1Z5 57345646 IC50 = 35800 nM T58093 C4GTE0 57345647 IC50 = 100100 nM T58093 CO8R3H 57878092 IC50 = 5 nM T58093 C0HY5X 57878097 IC50 = 2.3 nM T58093 C3W6PE 57878101 IC50 = 10 nM T58093 C2GJ1F 57878102 IC50 = 1.7 nM T58093 CX9UE4 57878122 IC50 = 1.6 nM T58093 C2F9SP 57878124 IC50 = 1.4 nM T58093 CH48QS 57878125 IC50 = 1.2 nM T58093 C5UJ7H 57878129 IC50 = 0.9 nM T58093 CU2KR4 57878131 IC50 = 1.7 nM T58093 C0WIY3 57878141 IC50 = 0.86 nM T58093 C1R5WU 57878145 IC50 = 1 nM T58093 C3XHZ9 70681653 IC50 = 1.3 nM T58093 C0C5BI 70685926 IC50 = 3.3 nM T58093 CMH5K3 70692221 IC50 = 2.3 nM T58093 C5SH2R 70694300 IC50 = 5.9 nM T58093 C5W1AK 138454269 IC50 = 2 nM T58093 CZUO38 155511087 IC50 = 2 nM T58093 C9F6LQ 155511457 IC50 = 5 nM T58093 C5DKE6 155511474 IC50 = 16 nM T58093 C45DSK 155512893 IC50 = 6 nM T58093 C6BQA2 155514815 IC50 = 11 nM T58093 CD58RH 155518934 IC50 = 5 nM T58093 C3WQH0 155520436 IC50 = 2 nM T58093 C0P4AY 155523706 IC50 = 10 nM T58093 CX3FD5 155526303 IC50 = 1 nM T58093 CEU4S5 155526689 IC50 = 0.63 nM T58093 CV3SG0 155529612 IC50 = 1 nM T58093 CJL2C8 155535353 IC50 = 18 nM T58093 CF5T2J 155536889 IC50 = 158 nM T58093 C7D4BJ 155541590 IC50 = 2 nM T58093 CL5AO7 155553287 IC50 = 20 nM T58093 CQF91W 155554205 IC50 = 3 nM T58093 CB1SN4 155557831 IC50 = 2 nM T58093 C94TBM 155560644 IC50 = 2 nM T58093 C4AD6J 155563341 IC50 = 1 nM T20600 D0J3SU 9847835 EC50 > 5000 nM T20600 C3T8NF 5288850 IC50 > 5000 nM T20600 C1KR5B 5327301 Ki = 22000 nM T20600 C37TKL 5327302 Ki = 1000 nM T20600 C64ZMN 5327304 Ki = 1400 nM T20600 C3IZ2W 5327307 Ki = 2300 nM T20600 C16DTL 5327308 Ki = 540 nM T20600 C4O3QY 5327309 Ki = 9700 nM T20600 C3GUM7 5327310 Ki = 2400 nM T20600 C3LZX9 8027611 IC50 > 20000 nM T20600 CFN2P6 9800285 Ki = 7500 nM T20600 CLTO67 9821317 IC50 = 18 nM T20600 C4XO3K 9821545 IC50 > 5000 nM T20600 CJI5T3 9823027 IC50 = 37 nM T20600 C74QTI 9823074 IC50 = 940 nM T20600 C6S3KT 9840223 Ki > 25000 nM T20600 CD05OL 9867192 IC50 = 1500 nM T20600 C2DMG1 9914167 IC50 > 5000 nM T20600 C9CV0Y 10001828 IC50 = 940 nM T20600 CX67SZ 10826725 Ki = 1000 nM T20600 CDX7A4 10963183 Ki = 190 nM T20600 CM8O6L 11257152 IC50 = 50 nM T20600 C4F8DC 11444079 IC50 > 500000 nM T20600 CDT9G3 11467504 IC50 = 3.44 nM T20600 CV4CP9 11496333 IC50 > 5000 nM T20600 CGE2J0 11497112 IC50 > 5000 nM T20600 C6IS9K 11509289 IC50 > 5000 nM T20600 C6L2MY 11509300 IC50 > 5000 nM T20600 CC31QO 11509301 IC50 > 5000 nM T20600 CS8OX7 11510566 IC50 > 500000 nM T20600 C7FY9B 11512139 IC50 > 5000 nM T20600 C15VFG 11515586 IC50 > 500000 nM T20600 CW6PC0 11519268 IC50 > 5000 nM T20600 CZC5D9 11525874 IC50 > 5000 nM T20600 C5BNE1 11533326 IC50 > 5000 nM T20600 CDK3Z5 11533935 IC50 = 3700 nM T20600 C4IC7E 11541867 IC50 > 500000 nM T20600 C3USR9 11543714 IC50 = 283 nM T20600 C3P2GZ 11548424 IC50 > 500000 nM T20600 CVX4M6 11548909 EC50 > 5000 nM T20600 C17OJS 11572844 IC50 = 201 nM T20600 CF0V3P 11576540 IC50 > 5000 nM T20600 C1T9DY 11576622 IC50 > 5000 nM T20600 C03KPR 11576852 EC50 > 5000 nM T20600 CN67DR 11583840 IC50 > 5000 nM T20600 CPD0M8 11584106 IC50 > 5000 nM T20600 CL16IM 11591540 IC50 > 5000 nM T20600 CE2TX6 11591919 IC50 > 500000 nM T20600 CG4Z9A 11598106 IC50 > 10000 nM T20600 CV6MF1 11614728 IC50 > 500000 nM T20600 CFP19E 11619968 IC50 > 5000 nM T20600 CA0LH6 11624920 IC50 > 5000 nM T20600 CEY39D 11628992 IC50 > 500000 nM T20600 C6UAV3 11632008 IC50 = 216 nM T20600 C6Y5MG 11634372 IC50 > 5000 nM T20600 CKJE92 11634649 IC50 > 5000 nM T20600 C91JNO 11639020 IC50 = 124 nM T20600 C4MCW2 11646889 IC50 = 137 nM T20600 C2KFU3 11647018 IC50 > 5000 nM T20600 CH20JE 11652994 IC50 = 2850 nM T20600 CN32TX 11664423 IC50 > 500000 nM T20600 CUD05C 11670894 IC50 > 5000 nM T20600 CX97NT 11684618 IC50 > 5000 nM T20600 C05YRV 11699954 IC50 > 500000 nM T20600 CKEX64 11700402 IC50 > 500000 nM T20600 C89COT 11705942 IC50 > 5000 nM T20600 C86PAH 11712912 IC50 > 5000 nM T20600 CXH9M5 16749067 IC50 = 407 nM T20600 C2DJ5W 16749068 IC50 = 9550 nM T20600 COM07G 16749069 IC50 = 698 nM T20600 CPG8Q0 16749161 IC50 = 744 nM T20600 CG84TK 16749162 IC50 = 823 nM T20600 CT3HD1 16749163 IC50 = 650 nM T20600 CZM4X2 16749164 IC50 = 610 nM T20600 CUZ8N4 16749267 IC50 = 8900 nM T20600 CMEK96 16749268 IC50 = 5025 nM T20600 C01HBN 16749269 IC50 = 918 nM T20600 CWG3C8 16749270 IC50 = 840 nM T20600 C8R3GD 16749271 IC50 = 515 nM T20600 CTI80F 25178948 EC50 > 5000 nM T20600 C2GI4J 25178949 EC50 > 5000 nM T20600 CQ2GM9 25178950 EC50 > 5000 nM T20600 C4GFV6 25179140 EC50 > 5000 nM T20600 CYL36B 25179141 IC50 = 4425 nM T20600 CGC69Q 25179143 EC50 > 5000 nM T20600 C27YJF 25179144 IC50 = 9967 nM T20600 C2YTB7 25179145 EC50 > 5000 nM T20600 C6GTV3 25179324 EC50 > 5000 nM T20600 CIC46T 25179513 EC50 > 5000 nM T20600 CK96WB 25179514 EC50 > 5000 nM T20600 CGX78D 25217029 IC50 = 450 nM T20600 CW2L9Q 25217030 IC50 = 770 nM T20600 C8UTC4 25217031 IC50 = 509 nM T20600 CZ43KQ 25217032 IC50 = 927 nM T20600 C2P9NI 25217145 IC50 = 4930 nM T20600 C8C9XU 42618276 IC50 > 15000 nM T20600 CFO93N 42618277 IC50 = 12833 nM T20600 CS1KQ0 42618278 IC50 = 325 nM T20600 CVI16X 42618279 IC50 = 545 nM T20600 C3MRA0 42618280 IC50 = 568 nM T20600 C8UO9S 42618281 IC50 = 425 nM T20600 C68NPR 42618282 IC50 = 453 nM T20600 CL41SD 42618283 IC50 = 591.7 nM T20600 CJ7U2E 42618284 IC50 = 151 nM T20600 CZL8C7 42618285 IC50 = 188 nM T20600 CNIQ28 42618286 IC50 = 230 nM T20600 C91OMB 42618287 IC50 = 9833 nM T20600 C5AC1L 42618288 IC50 = 156 nM T20600 CFU5T2 42618289 IC50 = 197 nM T20600 CK9H3M 42618290 IC50 = 280 nM T20600 CV4H2J 42618291 IC50 = 241 nM T20600 C7VPU3 42618292 IC50 = 358 nM T20600 C6R2FM 42618293 IC50 = 468 nM T20600 CT7VO2 44157085 IC50 > 500000 nM T20600 CWMU91 44157086 IC50 > 500000 nM T20600 C6LZ5Y 44157087 IC50 > 500000 nM T20600 CYSJ79 44157089 IC50 > 500000 nM T20600 CMX7W1 44157090 IC50 > 500000 nM T20600 C7B3VE 44158086 IC50 > 500000 nM T20600 C20WEJ 44158089 IC50 > 500000 nM T20600 C68KOD 44158154 IC50 > 500000 nM T20600 C4C1RU 44158155 IC50 > 500000 nM T20600 CN1YR9 44158157 IC50 > 500000 nM T20600 C80XPD 44158237 IC50 > 500000 nM T20600 CN09UV 44158238 IC50 > 500000 nM T20600 CT9DF4 44158240 IC50 > 500000 nM T20600 CHDF62 44158242 IC50 > 500000 nM T20600 CS6X1C 44158325 IC50 > 500000 nM T20600 C17TEZ 44158326 IC50 > 500000 nM T20600 CZ0VT3 44158328 IC50 > 500000 nM T20600 CD8WB9 44304162 Ki = 57000 nM T20600 CAB39E 44331552 IC50 = 32400 nM T20600 CE0FW4 44331565 IC50 = 21400 nM T20600 C8SZN9 44331566 IC50 = 12000 nM T20600 CMFW61 44331567 IC50 = 22600 nM T20600 CHYL38 44331577 IC50 = 1620 nM T20600 C1I9QH 44331578 IC50 = 18900 nM T20600 C4VGZ1 44331579 IC50 = 10100 nM T20600 CRZ01H 44331580 IC50 = 20500 nM T20600 CFOR90 44331674 IC50 = 14500 nM T20600 CK7VI8 44331675 IC50 = 717 nM T20600 CH7GS4 44331676 IC50 > 50000 nM T20600 C4FOD3 44331693 IC50 > 50000 nM T20600 CJY5L2 44331739 IC50 = 28600 nM T20600 C8N2GQ 44331740 IC50 = 11800 nM T20600 CW9K4Q 44331815 IC50 = 3370 nM T20600 CT76DG 44331816 IC50 = 33400 nM T20600 CC70GF 44331830 IC50 = 2530 nM T20600 CNJ19L 44331876 IC50 = 11110 nM T20600 C46IPA 44331879 IC50 > 10000 nM T20600 CP0Y8M 44331898 IC50 = 10 nM T20600 CF3R6W 44331908 IC50 > 10000 nM T20600 CTM5W1 44331914 IC50 = 3.5 nM T20600 C0YZ9O 44331915 IC50 = 15 nM T20600 C4NK1S 44331942 IC50 = 10 nM T20600 CXKY19 44331943 IC50 = 18560 nM T20600 C3FC8D 44331944 IC50 > 10000 nM T20600 CH1ZF2 44331953 IC50 = 589 nM T20600 C0QJ8V 44331957 IC50 = 4600 nM T20600 C1HBX6 44331963 IC50 = 14030 nM T20600 C7UXK5 44331964 IC50 = 10000 nM T20600 C42PGN 44331965 IC50 = 308 nM T20600 C5J7KX 44331966 IC50 > 50000 nM T20600 CG83FS 44331967 IC50 = 12500 nM T20600 CGAJ95 44331977 IC50 = 3610 nM T20600 CCYX84 44331980 IC50 > 10000 nM T20600 C5UIO2 44331987 IC50 = 32500 nM T20600 C0PM5C 44332004 IC50 = 4180 nM T20600 C4ENB1 44332005 IC50 = 1010 nM T20600 CFK4Z1 44332024 IC50 = 1280 nM T20600 CTM3G2 44332026 IC50 = 2720 nM T20600 C48ZEW 44332028 IC50 > 50000 nM T20600 C30MKG 44332029 IC50 > 50000 nM T20600 C7OS9X 44332050 IC50 = 9750 nM T20600 C9Y6NP 44332051 IC50 = 5050 nM T20600 C0VGF8 44332058 IC50 = 5860 nM T20600 CQU84D 44332068 IC50 = 21200 nM T20600 CBL91D 44332078 IC50 = 51200 nM T20600 C4VCM3 44332093 IC50 = 5900 nM T20600 C92QVT 44332108 IC50 = 1430 nM T20600 CQLZ09 44332109 IC50 = 13800 nM T20600 C4CUL6 44332112 IC50 = 3030 nM T20600 CN2YM6 44332113 IC50 = 1900 nM T20600 C4CY8K 44332118 IC50 = 7000 nM T20600 CXZ2N1 44332120 IC50 = 42700 nM T20600 CD56PK 44332121 IC50 > 50000 nM T20600 C5A6OJ 44332128 IC50 = 14500 nM T20600 C6IZ2R 44332129 IC50 = 3160 nM T20600 C5DY0G 44332136 IC50 = 1430 nM T20600 CQ1K9H 44332311 IC50 = 37 nM T20600 C9LOS2 44332330 IC50 = 305 nM T20600 C2U6GB 44332331 IC50 = 10300 nM T20600 CH01QW 44332332 IC50 = 11800 nM T20600 C8D5TB 44364680 Ki = 120 nM T20600 CJ6QG4 44417479 IC50 > 500000 nM T20600 C7RX9I 44418960 Ki = 550000 nM T20600 CXR1V5 44434249 IC50 = 61 nM T20600 C8Z4WO 44459967 IC50 = 5128.61 nM T20600 C86ORE 44459987 IC50 = 3548.13 nM T20600 CDY2W5 49796910 IC50 = 1.7 nM T20600 C3M2BW 52918163 IC50 = 8700 nM T20600 CF24IM 52918177 IC50 = 6900 nM T20600 CR9I7F 52918178 IC50 = 13450 nM T20600 C2VPU1 52918179 IC50 = 7750 nM T20600 C8Z2TQ 54580470 IC50 > 10000 nM T20600 CMU0B4 54581481 IC50 > 10000 nM T20600 CCS8Y3 54581987 IC50 = 1165 nM T20600 CJEP38 54582484 IC50 = 7666 nM T20600 C61NWL 54582924 IC50 = 9125 nM T20600 CO0AG3 54583923 IC50 = 747 nM T20600 CI2DL4 54583924 IC50 = 3475 nM T20600 CV2WU1 54583925 IC50 = 4700 nM T20600 CXA51D 54584867 IC50 = 6950 nM T20600 C8YSL0 54585834 IC50 = 1012 nM T20600 C9B5OF 54586343 IC50 = 2987 nM T20600 C7A8ER 54587376 IC50 = 9200 nM T20600 CGY3W2 71471109 IC50 > 100000 nM T20600 CKZ2H0 71582971 IC50 > 500000 nM T20600 C4WJ5F 71582972 IC50 > 500000 nM T20600 CXA62J 71582973 IC50 = 1030 nM T20600 CNZS31 71582974 IC50 > 500000 nM T20600 CE4L9D 71582975 IC50 > 500000 nM T20600 CXMS80 71583078 IC50 > 500000 nM T20600 C30UIL 71583079 IC50 > 500000 nM T20600 CJBC14 71583080 IC50 = 2610 nM T20600 C57MOP 71583081 IC50 > 500000 nM T20600 CS0YK9 71583082 IC50 > 500000 nM T20600 C3UTO9 71583083 IC50 > 500000 nM T20600 CW1R5Q 71583084 IC50 > 500000 nM T20600 CR57LS 71583192 IC50 > 500000 nM T20600 C8B3NZ 71583193 IC50 > 500000 nM T20600 CB6DY7 71583194 IC50 > 500000 nM T20600 CANH70 71716242 IC50 > 100000 nM T20600 C40WIR 71718085 IC50 = 100000 nM T20600 CU75VK 71719897 IC50 = 600 nM T20600 CBV6F1 71720507 IC50 > 100000 nM T20600 C4U5TO 76311196 IC50 > 10000 nM T20600 CSI53E 76311200 IC50 > 10000 nM T20600 CNOL37 76311201 IC50 = 3878 nM T20600 C8IS5Q 76314800 IC50 = 5082 nM T20600 CK41QI 76314804 IC50 > 10000 nM T20600 CHS61N 76314805 IC50 > 10000 nM T20600 CDY7K0 76318413 IC50 = 3790 nM T20600 CB2N6G 76322078 IC50 > 10000 nM T20600 C8SPW6 76322082 IC50 > 10000 nM T20600 CC2EP6 76325698 IC50 > 10000 nM T20600 CFY79U 76332916 IC50 > 10000 nM T20600 CD35SI 76332917 IC50 > 10000 nM T20600 C3FQX0 76336535 IC50 > 10000 nM T20600 CV4PE6 76336536 IC50 > 10000 nM T20600 CKCI60 90663142 IC50 = 310 nM T20600 C3GPO7 118723314 IC50 = 500000 nM T20600 C8H0EL 118723315 IC50 = 28500 nM T20600 CTE1O2 118723316 IC50 = 500000 nM T20600 CE8O9P 118723317 IC50 = 500000 nM T20600 C48DEF 118723325 IC50 = 500000 nM T20600 C67QMY 118723326 IC50 = 500000 nM T20600 CCJ27M 118723327 IC50 = 500000 nM T20600 COG92V 118723328 IC50 = 500000 nM T20600 CSX85P 118723329 IC50 = 500000 nM T20600 CICB42 118723330 IC50 = 78900 nM T20600 C13BRQ 118723331 IC50 = 12900 nM T20600 CWM2E8 133081971 IC50 > 9999 nM T20600 D08ORM 15487887 IC50 = 8 nM T20600 D0N5MU 4117381 Ki > 50000 nM T20600 D0Q9XX 515950 Ki = 1700 nM T20600 D0V6DX 10640 IC50 = 474 nM T20600 D0Y5IQ 44255320 IC50 = 5000 nM T28330 D04JEE 4946 EC50 > 5011.87 nM T28330 D0H7FW 9870520 Ki = 28.84 nM T28330 D0LI1C 44469321 IC50 > 30000 nM T28330 D01ZXW 122077 IC50 = 0.5623 nM T28330 D0C8ZD 121964 IC50 = 1900 nM T28330 D0EG1F 9914672 Ki = 79.43 nM T28330 D0F6CT 51353551 EC50 = 0.0024 nM T28330 D0W8TS 9898185 IC50 = 3162.28 nM T28330 D0W9ZY 52949124 EC50 = 0.5248 nM T28330 D0XJ0S 108187 IC50 = 1047.13 nM T28330 C7YKF2 1098327 Ki < 10000 nM T28330 CR7Y4G 1109919 Ki > 10000 nM T28330 CA0XN1 3081599 EC50 = 28 nM T28330 CF74HA 6918156 IC50 = 0.5 nM T28330 C6E0TB 9832467 Ki < 10000 nM T28330 C07OFK 9892971 IC50 > 10000 nM T28330 C57IBS 9913081 Ki < 10000 nM T28330 CRT68S 9960432 Ki = 125.89 nM T28330 CKTR60 10008654 IC50 = 5.2 nM T28330 CV56TJ 10031013 IC50 = 75.86 nM T28330 CD7XO3 10032955 EC50 = 3.162 nM T28330 C7SQA8 10032956 IC50 = 229.09 nM T28330 CDT69G 10051431 IC50 = 440 nM T28330 CFO8L6 10071178 Ki = 31.62 nM T28330 CL8M2B 10320262 Ki = 25.12 nM T28330 C16YAW 10343558 Ki = 25.12 nM T28330 CM1D3V 10350069 IC50 = 724.44 nM T28330 C4DIK2 10366068 Ki = 25.12 nM T28330 CD6B7H 10373077 EC50 = 3.981 nM T28330 CTE7N2 10388627 Ki = 25.12 nM T28330 CA5B8O 10391834 IC50 = 1584.89 nM T28330 CYU58T 10415786 IC50 = 39.81 nM T28330 C5Z8IP 10433726 Ki = 25.12 nM T28330 CM97BA 10460632 Ki = 3006 nM T28330 CB1X4K 10483574 IC50 = 79.43 nM T28330 CVE86S 10507071 IC50 = 6850 nM T28330 C91ZVY 10507109 Ki = 50.12 nM T28330 C36HIS 10507561 IC50 = 15.85 nM T28330 CKY68B 10509945 EC50 = 9.12 nM T28330 C1AE8J 10531224 IC50 = 1318.26 nM T28330 C9SUK0 10531430 IC50 = 1584.89 nM T28330 C4S2YR 10555164 IC50 = 138.04 nM T28330 CJZ47Q 10555363 IC50 = 36.31 nM T28330 CRI50M 10555571 IC50 = 42.66 nM T28330 CIN1C4 10555804 IC50 = 13.8 nM T28330 CM7LP6 10556460 IC50 = 309.03 nM T28330 C6LR2W 10580108 IC50 = 389.05 nM T28330 C0IT5X 10603713 IC50 = 17.38 nM T28330 CBRX06 10603714 IC50 = 20.89 nM T28330 C0AV6Q 10626596 IC50 = 524.81 nM T28330 CG02LF 10627173 IC50 = 10.81 nM T28330 CWF78P 10649606 EC50 = 0.014 nM T28330 C1QT8S 10674604 IC50 = 891.25 nM T28330 CXZ4C9 10675328 IC50 = 14.45 nM T28330 C84WOB 10698051 IC50 = 87.1 nM T28330 C89BME 10698109 IC50 = 154.88 nM T28330 CX8P5U 10698905 IC50 = 29.51 nM T28330 C90UHA 10699165 IC50 = 660.69 nM T28330 CG1KP5 10700916 EC50 = 1.549 nM T28330 CN53KG 10721792 IC50 = 120.23 nM T28330 C3R0HF 10722103 IC50 = 112.2 nM T28330 CA9O7Y 10722372 IC50 = 2511.89 nM T28330 CHD26N 10746778 IC50 = 1995.26 nM T28330 C7MS8F 10769675 IC50 = 478.63 nM T28330 C7KR4C 10769902 IC50 = 13.18 nM T28330 CU8KV7 10770092 IC50 = 17.78 nM T28330 CU59WT 10793168 IC50 = 107.15 nM T28330 CLMG75 10793883 IC50 = 38.9 nM T28330 C4G5HX 10794311 IC50 > 10000 nM T28330 CV2LI6 10817241 IC50 = 128.82 nM T28330 C8VBP1 10817395 IC50 = 8.318 nM T28330 CNL17K 10817407 IC50 = 354.81 nM T28330 CPER12 10819755 EC50 = 0.02512 nM T28330 C25UOS 10841112 IC50 = 89.13 nM T28330 C3Y6WE 10841358 IC50 = 42.66 nM T28330 C0ODR4 11027990 IC50 = 35.2 nM T28330 CT7HI5 11154873 Ki > 10000 nM T28330 CGR9A8 11178846 Ki > 10000 nM T28330 C2O3XT 11202178 Ki > 10000 nM T28330 C3NCV9 11212985 Ki > 10000 nM T28330 C8WK7R 11248998 Ki < 10000 nM T28330 C72OIE 11259485 Ki < 10000 nM T28330 CVL2X8 11281656 Ki > 10000 nM T28330 C2ZUE8 11292979 Ki < 10000 nM T28330 CL38VT 11293780 Ki < 10000 nM T28330 CD4I0A 11305046 Ki > 10000 nM T28330 CKL0X6 11316421 Ki < 10000 nM T28330 CBNS24 11316813 Ki < 10000 nM T28330 C9VA4Z 11352971 Ki > 10000 nM T28330 CU75AT 11353036 Ki < 10000 nM T28330 C3QE5S 11362975 Ki > 10000 nM T28330 COG3H2 11363465 Ki > 10000 nM T28330 C9DF4G 11363566 Ki < 10000 nM T28330 CXH69E 11385416 Ki > 10000 nM T28330 C9IX1T 11396307 Ki > 10000 nM T28330 CRA51C 11420366 Ki < 10000 nM T28330 COSZ16 11430523 Ki < 10000 nM T28330 CT0RI9 11431264 Ki < 10000 nM T28330 CXIN31 11442229 Ki > 10000 nM T28330 C9U8VO 11453391 Ki < 10000 nM T28330 C6AYO0 11454197 Ki < 10000 nM T28330 CE96SJ 11464858 Ki > 10000 nM T28330 C58JUC 11465671 Ki < 10000 nM T28330 CF9U1W 11511721 Ki = 1174.9 nM T28330 CV02EM 11512151 Ki = 50.12 nM T28330 C9TE6V 11527738 Ki = 10000 nM T28330 CYF52S 11534407 Ki = 79.43 nM T28330 C21ELY 11534594 Ki = 31.62 nM T28330 CA8WL2 11541048 Ki = 63.1 nM T28330 C7QYJ1 11555166 Ki = 724.44 nM T28330 C16KZS 11556194 Ki = 501.19 nM T28330 C8B2SH 11584582 Ki = 79.43 nM T28330 CK4H5O 11584903 Ki = 8709.64 nM T28330 C24OIW 11592162 Ki < 10000 nM T28330 CN6AR3 11605814 Ki < 10000 nM T28330 CT29GZ 11613982 Ki < 10000 nM T28330 CO3F1P 11627917 Ki = 79.43 nM T28330 C4EHB7 11635377 Ki = 12.59 nM T28330 COM97A 11656338 Ki = 5888.44 nM T28330 C51UDK 11667741 IC50 = 8100 nM T28330 CW79UI 11693225 Ki = 199.53 nM T28330 C42YZA 11700410 Ki = 158.49 nM T28330 CV9M3K 11712880 Ki = 1513.56 nM T28330 CK4SG5 11754311 Ki = 25.12 nM T28330 C65DTB 11765552 IC50 = 60.26 nM T28330 CSX23A 11786290 Ki < 10000 nM T28330 C8L2NZ 11801335 IC50 = 100 nM T28330 CSH7X6 11801911 IC50 = 16.98 nM T28330 C30NLE 15002730 Ki = 25.12 nM T28330 C2LBG8 15002734 Ki = 25.12 nM T28330 C5I4LT 15667001 IC50 = 16 nM T28330 CDJF92 15667003 IC50 = 4.2 nM T28330 CXH92N 15667011 IC50 = 0.99 nM T28330 C6QDI1 16090646 Ki < 10000 nM T28330 C3UCY1 16090647 Ki < 10000 nM T28330 C3HO2S 16090649 Ki < 10000 nM T28330 C4FKT8 16090650 Ki < 10000 nM T28330 CB19JY 16090651 Ki < 10000 nM T28330 CW7KL5 16090652 Ki > 10000 nM T28330 C9Q5YA 16090653 Ki > 10000 nM T28330 CA4PD3 16090658 Ki > 10000 nM T28330 CY9MB5 16090684 Ki > 10000 nM T28330 CY91OD 16090685 Ki > 10000 nM T28330 C4P8KS 16090686 Ki < 10000 nM T28330 C17IOA 16090687 Ki > 10000 nM T28330 C4ETX5 16090688 Ki > 10000 nM T28330 C37DEW 16090689 Ki > 10000 nM T28330 C7Q8LP 16090690 Ki > 10000 nM T28330 COJ46W 16090691 Ki < 10000 nM T28330 CNSU17 16090692 Ki > 10000 nM T28330 C49PFE 16090693 Ki > 10000 nM T28330 CI0XC5 16090694 Ki > 10000 nM T28330 C6QDP7 16090695 Ki > 10000 nM T28330 C3AVH8 16090699 Ki = 3162.28 nM T28330 C9R2PB 16090700 Ki = 199.53 nM T28330 C9K8RC 16090701 Ki = 7943.28 nM T28330 CH1UB0 16090702 Ki = 1995.26 nM T28330 CD7S4Q 16090703 Ki > 10000 nM T28330 CRS7B1 16090773 Ki > 10000 nM T28330 C2KCS0 16090774 Ki > 10000 nM T28330 C8IGT2 16090780 Ki > 10000 nM T28330 CM72TB 16090781 Ki > 10000 nM T28330 C8CI1X 16090782 Ki < 10000 nM T28330 C9QGU2 16090783 Ki > 10000 nM T28330 CF2IW8 16090784 Ki < 10000 nM T28330 CKCX80 16090785 Ki > 10000 nM T28330 C3D8HU 16090786 Ki < 10000 nM T28330 C8WSC9 16090788 Ki > 10000 nM T28330 CYQP41 16090789 Ki = 2511.89 nM T28330 C6MV4D 16090790 Ki > 10000 nM T28330 CJ94QO 16090791 Ki > 10000 nM T28330 C2G8TD 16090792 Ki < 10000 nM T28330 CRF40D 16090793 Ki < 10000 nM T28330 CX68OS 16090794 Ki > 10000 nM T28330 C0V8WI 16090795 Ki < 10000 nM T28330 C06QBM 16090796 Ki < 10000 nM T28330 C5NER1 16090797 Ki < 10000 nM T28330 C3T9MH 16100406 Ki = 130 nM T28330 CH6F0V 16100408 Ki = 8300 nM T28330 CY5F4S 16162108 EC50 = 269.15 nM T28330 C7YG3M 16731537 Ki < 10000 nM T28330 C7U3FA 16731711 Ki = 371.54 nM T28330 C3G0VB 16731712 Ki < 10000 nM T28330 CD9KY3 16731870 Ki < 10000 nM T28330 C6RS1M 16731872 Ki < 10000 nM T28330 CQ45MJ 16731874 Ki > 10000 nM T28330 C8FH9C 16732017 Ki = 6456.54 nM T28330 C9I7PZ 16732018 Ki = 4073.8 nM T28330 C8JR5Q 16732019 Ki = 1737.8 nM T28330 C2OQ0S 16732020 Ki = 6456.54 nM T28330 C5VUZ7 16732021 Ki = 389.05 nM T28330 CXN1C3 16732022 Ki < 10000 nM T28330 C34EYO 16732162 Ki = 457.09 nM T28330 C6CF0K 16732163 Ki < 10000 nM T28330 C4GZY1 16732164 Ki = 549.54 nM T28330 C8DU5M 16732165 Ki = 2511.89 nM T28330 CB7X3W 16732442 Ki < 10000 nM T28330 CY57CK 16732443 Ki = 5754.4 nM T28330 CO95FT 16732444 Ki = 2137.96 nM T28330 CE9M8H 16732592 Ki = 8128.31 nM T28330 C3J2CB 16732593 Ki = 6918.31 nM T28330 CU2FT3 16732598 Ki < 10000 nM T28330 CFT09X 16732750 Ki < 10000 nM T28330 CM4P7G 16732753 Ki < 10000 nM T28330 C9K4UR 16732755 Ki = 7943.28 nM T28330 CB2JR3 16732909 Ki > 10000 nM T28330 CZ14YT 16732911 Ki = 645.65 nM T28330 C35MZK 16732916 Ki = 1905.46 nM T28330 CR0A7J 16733051 Ki = 2951.21 nM T28330 C3LUI7 16733057 Ki < 10000 nM T28330 C9FU1Q 16733182 Ki < 10000 nM T28330 C93FYR 16733185 Ki = 549.54 nM T28330 CF3I5J 16733307 Ki = 660.69 nM T28330 CUF2R0 16733462 Ki = 8511.38 nM T28330 C0RH7Y 16733466 Ki = 2511.89 nM T28330 C1XWA0 16733469 Ki = 2089.3 nM T28330 CK04YG 16733644 Ki = 1698.24 nM T28330 C1RC2P 16733790 Ki < 10000 nM T28330 C76HVW 16755781 EC50 = 0.094 nM T28330 CO7F1T 16755782 EC50 = 1.1 nM T28330 CILG48 21842317 IC50 = 111 nM T28330 CLTI86 21842327 IC50 = 1200 nM T28330 C3NT8C 21842331 IC50 = 480 nM T28330 C53MSQ 21842340 IC50 = 293 nM T28330 CK8GY0 21842400 IC50 = 720 nM T28330 CPQ3K5 22171012 Ki = 25.12 nM T28330 C6VR4P 22171037 Ki = 25.12 nM T28330 C4Y3DN 22171039 Ki = 25.12 nM T28330 CH4V5J 22171089 Ki = 25.12 nM T28330 CKA98D 22171092 Ki = 25.12 nM T28330 CFL43N 23652473 IC50 > 1000000 nM T28330 CZ2PW8 24769543 EC50 = 0.033 nM T28330 CA7XZ6 24769546 IC50 = 0.018 nM T28330 C2YDQ3 24769604 IC50 = 0.01 nM T28330 CO46AU 24769605 EC50 = 0.065 nM T28330 CSCY65 24784940 IC50 = 2.5 nM T28330 C7HSF9 24784941 IC50 = 2.3 nM T28330 C14APO 24784942 IC50 = 22 nM T28330 C6X5AL 24785176 IC50 = 43 nM T28330 C4S1BJ 24785177 IC50 = 6.9 nM T28330 CE32FM 24785178 IC50 = 1.9 nM T28330 C6Y0AR 24785179 EC50 = 7.4 nM T28330 C0O2KU 24785180 EC50 = 5.5 nM T28330 C6ZNQ8 24785430 IC50 = 30 nM T28330 CXH90U 24785431 IC50 = 1.9 nM T28330 CC9TD5 24785432 EC50 = 175 nM T28330 C8A3XU 24785703 EC50 = 1.9 nM T28330 CZ14DY 24785705 IC50 = 0.42 nM T28330 CC8IW7 24861060 IC50 = 0.04 nM T28330 CZ9AS2 24861113 EC50 = 0.048 nM T28330 C6TM1P 24861114 EC50 = 0.053 nM T28330 C39NSA 24861174 EC50 = 0.4 nM T28330 CM0Q9T 24861391 IC50 = 0.03 nM T28330 CA5WE4 24861392 EC50 = 0.14 nM T28330 CCN34R 24861394 EC50 = 0.077 nM T28330 C5C4QR 24990933 IC50 < 50 nM T28330 C8HMZ0 25032312 Ki < 10000 nM T28330 C3NGL2 25032468 Ki < 10000 nM T28330 CK96SR 25033064 Ki < 10000 nM T28330 CM2Z9H 25033065 Ki < 10000 nM T28330 C1O7NJ 25033066 Ki < 10000 nM T28330 CITF86 25033148 Ki < 10000 nM T28330 C67SOQ 25033149 Ki < 10000 nM T28330 CJ10TY 25033150 Ki < 10000 nM T28330 C19WBD 44215880 Ki = 3.9 nM T28330 C6J7EK 44303510 IC50 > 10000 nM T28330 CWKM16 44303511 IC50 = 36.7 nM T28330 CY5Q8R 44303654 IC50 = 2175 nM T28330 CNH0W1 44303663 IC50 > 10000 nM T28330 CD80VI 44303664 IC50 = 2700 nM T28330 C0L8GD 44303722 IC50 = 364 nM T28330 CA8Z0J 44304324 IC50 = 190 nM T28330 C1VM8Q 44306360 IC50 = 31.62 nM T28330 C3ZDK0 44306744 IC50 = 19.95 nM T28330 CB5Q6O 44306823 IC50 = 5.012 nM T28330 CG9HF2 44306868 IC50 = 100 nM T28330 CP92WE 44306887 IC50 = 63.1 nM T28330 CN0SR5 44306888 IC50 = 100 nM T28330 C3MR8J 44328894 Ki = 10 nM T28330 C10ORA 44328951 Ki = 50.12 nM T28330 CZFL34 44329156 Ki = 79.43 nM T28330 CT7I5W 44330874 IC50 = 5.3 nM T28330 C4G1WN 44336539 EC50 = 0.02 nM T28330 C4HYP6 44355590 Ki = 3330 nM T28330 CVO2G3 44355745 Ki = 1080 nM T28330 CMS4H1 44355747 Ki = 3900 nM T28330 C8VW0Y 44355787 Ki = 10000 nM T28330 CHAZ51 44365304 IC50 = 3162.28 nM T28330 CMV8Q7 44365359 IC50 = 251.19 nM T28330 C1RNC2 44365788 IC50 = 10 nM T28330 CTD71M 44367000 IC50 = 2500 nM T28330 CN8SF3 44379428 Ki = 3 nM T28330 C9TZV6 44398261 IC50 = 3.8 nM T28330 CD69PS 44408411 Ki = 1000 nM T28330 C7QV6M 44408483 Ki = 560 nM T28330 C96ELC 44408632 Ki = 840 nM T28330 CI26KP 44417427 Ki > 10000 nM T28330 C0CV9L 44417429 Ki < 10000 nM T28330 CNZ3I4 44417439 Ki < 10000 nM T28330 C5OI3W 44418923 Ki > 10000 nM T28330 C4UPR1 44418924 Ki = 10000 nM T28330 CWT4D8 44425005 Ki = 7079.46 nM T28330 C2PEJ5 44425006 Ki = 3981.07 nM T28330 C7R2IK 44444763 Ki = 25.12 nM T28330 C0C1JA 44444767 Ki = 25.12 nM T28330 C91GMK 44444777 Ki = 25.12 nM T28330 CL94GA 44451519 Ki = 446.68 nM T28330 CXJ5N0 44451522 Ki = 616.6 nM T28330 CN8B5I 44451523 Ki < 10000 nM T28330 CMF6V5 44451547 Ki = 2089.3 nM T28330 C2MP5A 44451581 Ki = 281.84 nM T28330 C9SC7M 44451622 Ki = 2344.23 nM T28330 CH1K6S 44451830 Ki < 10000 nM T28330 CWEV38 44451843 Ki = 3890.45 nM T28330 CIS9D2 44451877 Ki = 1548.82 nM T28330 CVN2E4 44451920 Ki = 2344.23 nM T28330 C4DL5C 44469677 IC50 = 1 nM T28330 C9HFJ2 44562296 EC50 = 0.097 nM T28330 C1UA9S 44562297 EC50 = 0.04 nM T28330 CWT26N 44562298 EC50 = 0.095 nM T28330 C42LFU 44562299 IC50 = 0.08 nM T28330 CK78HN 44562300 EC50 = 0.082 nM T28330 C3QH7F 44562301 IC50 = 0.016 nM T28330 CSJ76G 44562302 EC50 = 0.034 nM T28330 CZ1MF9 44562303 IC50 = 0.067 nM T28330 CQ72YB 44562304 EC50 = 0.074 nM T28330 C9CDJ6 44562305 IC50 = 0.24 nM T28330 CM8A3V 44562306 EC50 = 0.097 nM T28330 CS3C0V 44562307 EC50 = 0.1 nM T28330 CR5Y4S 44562308 EC50 = 0.21 nM T28330 C9APN5 44562309 EC50 = 0.16 nM T28330 CF1BD0 44562310 EC50 = 0.18 nM T28330 C2JL9N 44562311 EC50 = 0.77 nM T28330 CT57RP 44562312 EC50 = 0.097 nM T28330 C2Y5XD 44562313 EC50 = 0.46 nM T28330 CJ72VF 44562314 EC50 = 0.14 nM T28330 C3IB9C 44578251 EC50 = 74 nM T28330 C3HFG1 44578305 IC50 = 8 nM T28330 CQ1DN3 44578398 IC50 = 630 nM T28330 C5FA0D 44578399 EC50 = 9.1 nM T28330 CG5PO8 44578422 IC50 = 16 nM T28330 C97ZLF 44578423 IC50 = 1.9 nM T28330 C5X3RK 44578424 EC50 = 1.1 nM T28330 CCS0G8 44578455 IC50 = 8.6 nM T28330 C45QLM 44578456 EC50 = 106 nM T28330 CW0F5K 44578457 EC50 = 0.078 nM T28330 CV5X3L 44578529 EC50 = 962 nM T28330 C4U0QS 44578530 IC50 = 130 nM T28330 CB31ZF 44578531 EC50 = 1349 nM T28330 CB9X2L 44578562 EC50 = 471 nM T28330 C8ES9Z 44578611 IC50 = 35 nM T28330 C65UYX 44578647 IC50 = 1.9 nM T28330 C94RSO 44578686 EC50 = 0.25 nM T28330 CLW1R5 44578727 EC50 = 0.53 nM T28330 CDIW83 44578728 EC50 = 0.13 nM T28330 CCP04Y 44578729 EC50 = 0.12 nM T28330 CJE1O8 44578764 EC50 = 0.26 nM T28330 C2A4JT 44578767 IC50 = 0.45 nM T28330 CPV6Q1 44578772 EC50 = 308 nM T28330 C6FE1M 45102806 Ki = 158.49 nM T28330 CM6BH7 45255234 Ki = 251.19 nM T28330 CYTL70 45486933 Ki = 100 nM T28330 CQH80S 45486935 Ki = 251.19 nM T28330 C7YUL8 45486936 Ki = 158.49 nM T28330 C1KLB2 45486940 Ki = 1995.26 nM T28330 COT6U7 45486941 Ki = 398.11 nM T28330 CAQ7Z9 45486947 Ki = 199.53 nM T28330 C6FGL0 45486949 Ki = 3981.07 nM T28330 CSR39Z 45486955 Ki = 199.53 nM T28330 CDZ82O 45486958 Ki = 3162.28 nM T28330 CMI20Q 45486964 Ki = 398.11 nM T28330 CD02XL 45486967 Ki = 158.49 nM T28330 C1X3BW 45486968 Ki = 316.23 nM T28330 CC8W1B 45486969 Ki = 199.53 nM T28330 CV17ZB 45486970 Ki = 3981.07 nM T28330 CZ04GO 45486971 Ki > 10000 nM T28330 C2WJI9 45486974 Ki = 25.12 nM T28330 C5HP4B 45486976 Ki = 251.19 nM T28330 CXR7T6 45486985 Ki = 316.23 nM T28330 CIX0G1 45486994 Ki = 1000 nM T28330 C1PZ8J 45486995 Ki = 1995.26 nM T28330 C06PMK 45486997 Ki = 3981.07 nM T28330 CQ31XM 45487002 Ki = 125.89 nM T28330 C3YB8W 45487003 Ki = 79.43 nM T28330 C6SQZ7 45487006 Ki = 100 nM T28330 CGH4V3 46234820 IC50 = 80.1 nM T28330 C5KH7S 46234969 IC50 = 4.24 nM T28330 CQAS17 46234970 IC50 = 44.7 nM T28330 CD0WG8 46235271 EC50 = 0.1202 nM T28330 CHD2N7 46235272 EC50 = 2.7 nM T28330 C94EJG 46869398 EC50 = 0.063 nM T28330 C8Y2QS 49798104 Ki > 10000 nM T28330 C6LEM8 49798106 IC50 = 125.89 nM T28330 C8EG6Y 49798111 Ki = 1400 nM T28330 C24DUW 49798112 Ki = 9 nM T28330 C2US0X 52940616 EC50 = 522 nM T28330 C5T0BN 52942901 EC50 = 91.3 nM T28330 CCOU43 52943046 EC50 = 628 nM T28330 CS2DM8 52944224 EC50 = 160 nM T28330 CL5G9A 52945789 EC50 = 1810 nM T28330 CW60FV 52946666 EC50 = 645 nM T28330 C4QWB8 52946667 IC50 = 246 nM T28330 CP0NO1 52950956 IC50 > 700 nM T28330 C7PC2V 52950958 IC50 > 700 nM T28330 CMYU60 52951093 IC50 > 700 nM T28330 C8ZL7M 52951227 IC50 > 700 nM T28330 C2VK4G 52951333 IC50 > 700 nM T28330 CG80QW 52951789 IC50 > 700 nM T28330 CXZL73 52952034 IC50 > 700 nM T28330 C6UQ3N 53233689 EC50 = 0.065 nM T28330 C2DIE0 53465843 Ki = 973 nM T28330 CB90RU 53465844 Ki = 0.32 nM T28330 C9J3NZ 54580263 EC50 = 38 nM T28330 CN56CG 54580264 IC50 = 2925 nM T28330 C74EHP 54580265 EC50 = 286 nM T28330 CV4Z2K 54580266 IC50 = 2.4 nM T28330 C6WDJ8 54580267 EC50 = 61 nM T28330 CF0V5K 54580295 EC50 = 0.71 nM T28330 CE98TJ 54580296 EC50 = 17 nM T28330 CGP10T 54581259 IC50 > 10000 nM T28330 CK85VP 54581260 IC50 = 35 nM T28330 C0XN2Z 54581261 EC50 = 34 nM T28330 C4SC7B 54581301 EC50 = 41 nM T28330 C8YT9J 54581302 EC50 = 9.6 nM T28330 CXP3W9 54582287 EC50 = 6.1 nM T28330 C5NZ0G 54582288 EC50 = 37 nM T28330 C7MT8A 54582313 EC50 = 5020 nM T28330 C10GBP 54583260 EC50 = 1.8 nM T28330 CSD2T3 54583296 EC50 = 0.24 nM T28330 CF12HS 54583297 EC50 = 59 nM T28330 CK01LS 54583298 EC50 = 0.2 nM T28330 C40TZF 54584222 IC50 > 10000 nM T28330 COGN42 54584255 EC50 = 7.5 nM T28330 CW6E2U 54586147 IC50 = 35 nM T28330 CB7AL6 54586148 IC50 = 0.18 nM T28330 CF1M5T 54586149 IC50 = 174 nM T28330 C5ME1Z 54586174 IC50 = 16.9 nM T28330 CE5SJ2 54586175 IC50 = 9.9 nM T28330 C9XP0E 54587149 IC50 = 33 nM T28330 CZ9S1K 54587150 EC50 = 1.3 nM T28330 CT14KG 54587151 EC50 = 256 nM T28330 C4HMO9 56663037 IC50 > 700 nM T28330 CZL6U4 56663263 IC50 > 700 nM T28330 CRL92U 56666696 IC50 > 700 nM T28330 CV38BZ 56683899 IC50 > 700 nM T28330 CSX93Z 70681224 EC50 = 31.9 nM T28330 CP73WX 70683295 IC50 = 68.6 nM T28330 C9V7QF 70683305 IC50 = 87.6 nM T28330 C15FHQ 70685411 IC50 = 248 nM T28330 CCQ5U4 70689603 EC50 = 52.5 nM T28330 C7BJ3X 70689619 EC50 = 2116.8 nM T28330 CQXZ61 70691750 EC50 = 12.9 nM T28330 C07BDF 70693814 IC50 = 340 nM T28330 CCN89Z 70695922 EC50 = 400 nM T28330 C0IJ1E 70695933 IC50 = 373 nM T28330 CR6KF1 70695934 IC50 = 38.1 nM T28330 CWH6T3 72548703 IC50 = 0.12 nM T28330 CNC3S0 73345637 IC50 = 15000 nM T28330 C5KT3R 73346888 IC50 < 100000 nM T28330 CG2PW4 73348650 IC50 = 32 nM T28330 CYL21W 73348651 IC50 = 6450 nM T28330 CO8BC0 73350236 IC50 = 26660 nM T28330 CIFQ07 73350237 IC50 = 7460 nM T28330 C5G8NK 73350238 IC50 = 7200 nM T28330 CE17QO 73351737 IC50 = 26340 nM T28330 CEVU91 73353218 IC50 = 6940 nM T28330 CGSW23 73354720 IC50 = 24750 nM T28330 CA8MQ1 73354785 Ki = 15 nM T28330 C6C0SX 90663256 IC50 = 7400 nM T28330 CZ61LK 127034966 EC50 > 5011.87 nM T28330 CA0SN5 127034967 EC50 > 5011.87 nM T28330 C1GY2T 135156251 EC50 > 10000 nM T28330 C3ZNX5 135423404 Ki = 467.74 nM T28330 CR79SC 135529065 Ki = 117.49 nM T28330 C0OK8I 135610887 Ki = 588.84 nM T28330 CEX49M 136000594 EC50 = 88 nM T28330 C8IP3M 136036821 Ki = 72.44 nM T28330 C6EOV2 136036823 Ki = 316.23 nM T28330 CB89KA 155514270 EC50 = 0.2512 nM T28330 C9MB4S 155514432 EC50 = 0.2138 nM T28330 CDK7N6 155515427 EC50 = 0.3631 nM T28330 C07LPH 155516677 EC50 = 0.1288 nM T28330 CBJH23 155517239 IC50 = 0.1096 nM T28330 CB1SI3 155517761 EC50 = 0.5012 nM T28330 CBG5S4 155517868 EC50 = 912.01 nM T28330 CTV3M6 155521287 IC50 = 5940 nM T28330 CKC61A 155524181 EC50 = 0.06761 nM T28330 CH5AU4 155524770 EC50 = 0.1585 nM T28330 CAE58M 155526914 EC50 = 0.1622 nM T28330 C9HIR7 155530671 EC50 = 0.06026 nM T28330 C30VKS 155531277 EC50 = 11.75 nM T28330 CKL8Y2 155532425 EC50 = 0.1096 nM T28330 CN0VP5 155532759 IC50 = 0.1072 nM T28330 C12IEY 155533399 EC50 = 0.166 nM T28330 CVBR79 155533520 EC50 = 8.511 nM T28330 CHV1D9 155535107 EC50 = 0.1072 nM T28330 C09DZK 155535249 EC50 = 0.166 nM T28330 CNB7M5 155535579 EC50 = 0.1698 nM T28330 CKI3E1 155536333 EC50 = 0.1349 nM T28330 CO07KD 155537344 EC50 = 0.1072 nM T28330 C8QIH3 155539345 IC50 = 0.06026 nM T28330 C2FBL5 155540394 EC50 = 1.122 nM T28330 CWP54F 155540415 EC50 = 602.56 nM T28330 CMV82T 155540739 EC50 = 0.2455 nM T28330 CB18RV 155542488 EC50 = 0.1905 nM T28330 CGN96I 155542545 EC50 = 3.311 nM T28330 CY6E8B 155543163 EC50 = 0.2951 nM T28330 CS5N7E 155543846 EC50 = 0.9772 nM T28330 C39DSM 155543995 EC50 = 0.3715 nM T28330 C7K4ZA 155544674 EC50 = 0.1288 nM T28330 CLB1R7 155546692 EC50 = 0.3236 nM T28330 C7Z8OY 155547906 IC50 = 0.07943 nM T28330 C1PV3I 155548381 EC50 = 0.389 nM T28330 C1GEA7 155550911 EC50 = 1.622 nM T28330 CQ9S8X 155551968 EC50 = 0.2138 nM T28330 C1DG3Q 155552556 EC50 = 0.182 nM T28330 C4QSR2 155553269 IC50 = 40.74 nM T28330 C3K4NQ 155553502 EC50 = 11.75 nM T28330 C51ZHW 155555065 IC50 = 0.09772 nM T28330 C8V6RX 155555346 IC50 = 0.0871 nM T28330 CDF1E8 155557064 EC50 = 0.1148 nM T28330 CN68GS 155557285 EC50 = 229.09 nM T28330 CO1N8R 155558199 EC50 > 1000 nM T28330 C0GE9L 155559320 IC50 = 0.07586 nM T28330 C2DFE4 155560670 IC50 = 0.07943 nM T28330 CLI24D 155562281 IC50 = 0.04266 nM T28330 CFZ19O 155564367 EC50 = 117.49 nM T28330 CFYB81 155564421 EC50 = 0.1549 nM T28330 CQ8G9E 155566319 IC50 = 0.07413 nM T28330 CK98TD 155568312 EC50 = 0.5012 nM T28330 CP23WI 44572148 Ki = 173.78 nM T28330 D00OFV 3035433 IC50 = 1400 nM T28330 D01ADK 11693641 Ki > 10000 nM T28330 D01AQC 9811733 Ki = 3600 nM T28330 D02ZML 5311148 IC50 = 22.91 nM T28330 D03EPA 11051303 IC50 = 97.72 nM T28330 D05QBF 443375 Ki = 0.02344 nM T28330 D05RRZ 10348659 IC50 = 63.1 nM T28330 D05YZC 59751 Ki = 10.4 nM T28330 D06BRA 11520765 IC50 = 6456.54 nM T28330 D06CIH 11200806 IC50 = 4000 nM T28330 D06KWA 11442807 IC50 = 12700 nM T28330 D07ICW 11556976 Ki = 32 nM T28330 D07LQQ 11564210 Ki = 9.6 nM T28330 D09EMR 11136782 IC50 = 1949.84 nM T28330 D0E2OG 11614928 Ki = 910 nM T28330 D0F1VP 44409521 IC50 = 2800 nM T28330 D0F1XY 44408590 Ki > 10000 nM T28330 D0FF6S 16038374 IC50 > 2000 nM T28330 D0I8AF 9833444 EC50 = 0.04365 nM T28330 D0I9PH 16100409 Ki = 1900 nM T28330 D0J7GJ 44408484 Ki = 10000 nM T28330 D0N6DN 44408524 IC50 = 4073.8 nM T28330 D0O7PT 60182 IC50 = 195 nM T28330 D0QP2S 44408526 Ki = 1900 nM T28330 D0R4GI 11040230 Ki = 5100 nM T28330 D0S7SO 16100407 Ki > 10000 nM T28330 D0TR0U 10942040 IC50 = 1096.48 nM T28330 D0U6OA 10909103 Ki = 5700 nM T28330 D0V9DY 16100410 Ki = 7000 nM T28330 D0X7LC 11061906 Ki = 870 nM T28330 D0Z4SS 44572147 Ki = 3.715 nM T18143 D03VOJ 8768 IC50 = 239000 nM T18143 C54JUR 25043 IC50 = 141000 nM T18143 C70HVL 77888 IC50 = 137000 nM T18143 CPI2E4 80447 IC50 = 71600 nM T18143 C07AKH 786691 IC50 = 20000 nM T18143 CY4MC6 3505109 IC50 = 145000 nM T18143 CGN9J7 44267478 IC50 = 25000 nM T18143 CH4Q6A 145964401 IC50 = 6100 nM T18143 CHU61S 145964420 IC50 = 600 nM T18143 C6YCA8 145964710 IC50 = 700 nM T18143 CV6F7L 145966788 IC50 = 600 nM T18143 CBWX17 145967285 IC50 = 900 nM T18143 COR9X3 145972736 IC50 = 700 nM T18143 CQ0M2X 145972809 IC50 = 7500 nM T18143 CF95RZ 145972878 IC50 = 600 nM T18143 CXI0D1 145975081 IC50 = 700 nM T18143 CG84ZR 145975487 IC50 = 400 nM T18143 C91FOT 145976006 IC50 = 800 nM T18143 C3F4UH 145978039 IC50 = 500 nM T79062 D00TLN 2913 Ki = 50.12 nM T79062 D00XWD 135409453 Ki < 100 nM T79062 D01AZG 5073 Ki = 0.4 nM T79062 D01ZII 2726 Ki = 10.72 nM T79062 D02HED 4748 Ki = 23 nM T79062 D03ELL 2159 Ki = 25.12 nM T79062 D03WEX 9966051 Ki = 19 nM T79062 D04JEE 4946 EC50 > 5011.87 nM T79062 D05MBZ 129211 Ki = 84 nM T79062 D05XGO 11154555 Ki = 111 nM T79062 D05ZIK 4205 Ki = 265 nM T79062 D06XZR 27400 Ki = 25 nM T79062 D08VRO 3822 Ki = 1258.93 nM T79062 D09IOI 2170 Ki = 500 nM T79062 D09TPF 23897 Ki = 265 nM T79062 D0CQ0Z 33630 Ki = 280 nM T79062 D0D1AL 3559 Ki = 316.23 nM T79062 D0G8NN 119570 Ki = 1188 nM T79062 D0H3HM 60795 Ki = 10.3 nM T79062 D0H7KF 5002 Ki = 63.1 nM T79062 D0P0OU 11978813 Ki = 3.7 nM T79062 D0R1JV 60854 Ki = 5 nM T79062 D0R6RO 4184 Ki = 56 nM T79062 D0U1OE 5452 Ki = 70 nM T79062 D0UA0I 28693 Ki = 6.31 nM T79062 D0V4QS 135398745 Ki = 79.43 nM T79062 D0W5HK 216239 Ki = 7071 nM T79062 D0X6BV 6918314 Ki = 3900 nM T79062 D0Z1RV 135398737 Ki = 5.5 nM T79062 D0Z6UC 5358 Ki = 1000 nM T79062 D04GMY 11842633 Ki < 100 nM T79062 D08CJK 1150 Ki = 158.49 nM T79062 D09IRN 21071390 Ki = 8635 nM T79062 D0N1HW 5311200 Ki = 226.3 nM T79062 D0R9HI 11256720 Ki = 14230 nM T79062 D00OWF 5280953 Ki = 5500 nM T79062 D02JMI 9888211 Ki = 100 nM T79062 D03ZZH 9887537 Ki = 63.1 nM T79062 D06DZI 107780 Ki > 10000 nM T79062 D06ZVC 10150497 Ki = 679 nM T79062 D07BCO 5684 Ki = 10000 nM T79062 D08AWI 11430856 Ki = 700 nM T79062 D08PUW 64982 IC50 > 200000 nM T79062 D0B7SP 11292933 Ki = 158.49 nM T79062 D0K8NW 5074 Ki = 15.85 nM T79062 D0L9SN 4431 Ki = 0.6 nM T79062 D0M7LV 5761 Ki = 6.31 nM T79062 D0Q2JS 10436045 Ki = 63.1 nM T79062 D0U7VZ 11225102 Ki < 100 nM T79062 D0YP7L 6604889 Ki = 0.3388 nM T79062 CZUI83 2769 Ki = 1000 nM T79062 C5H9CN 9287 Ki = 102.33 nM T79062 CFGH18 27620 Ki = 364 nM T79062 C8Y6DE 37461 Ki = 63.1 nM T79062 C6WDL7 49756 Ki = 145 nM T79062 CIOE06 69729 Ki = 140 nM T79062 CN9GK1 104911 Ki > 10000 nM T79062 CBH8L0 156308 Ki = 5000 nM T79062 CGT8R0 160510 Ki = 280 nM T79062 CLK7P3 169713 IC50 = 143 nM T79062 C4J5ZF 185617 IC50 = 63400 nM T79062 C9XWA6 198914 Ki = 1100 nM T79062 CP2DY7 198967 Ki = 97000 nM T79062 CVI6X5 213046 Ki = 0.5 nM T79062 C2V5FA 398712 Ki = 30 nM T79062 CYV1R3 417052 Ki = 2960 nM T79062 CD8Z9H 424430 Ki = 26 nM T79062 C4O6RK 435595 Ki = 84 nM T79062 CFJ3R2 452533 Ki = 27 nM T79062 CGF6W2 642376 IC50 = 126600 nM T79062 CTN56Q 647533 Ki > 4000 nM T79062 CXQ6U0 735755 IC50 > 10000 nM T79062 C2VLP8 752521 Ki = 2083 nM T79062 C9FI5L 1296368 Ki = 25390 nM T79062 C6VZT7 1984087 Ki = 8000 nM T79062 CGS9R7 2133793 Ki = 4718 nM T79062 CG9N3A 2136365 Ki = 6371 nM T79062 CT8KN9 2232766 Ki = 2307 nM T79062 CA2OY6 2737389 Ki = 1.4 nM T79062 CE50LO 2756712 Ki = 25 nM T79062 C1C4LH 2843443 Ki = 12250 nM T79062 CRA6F5 2853434 Ki = 1473 nM T79062 C3QRD6 2867758 Ki = 6100 nM T79062 CL2G3H 2870750 Ki = 13020 nM T79062 CC74QS 2872937 Ki = 20090 nM T79062 CRF65H 2880253 Ki = 10100 nM T79062 CET7C8 2921525 Ki = 14100 nM T79062 C2DE6R 2927683 Ki = 3800 nM T79062 CF01YE 2928642 Ki = 8400 nM T79062 CY8R6Q 2948971 Ki = 18080 nM T79062 CLXQ01 2950739 Ki = 10400 nM T79062 CO0C7J 2962174 Ki = 84500 nM T79062 CAM8H3 3066250 IC50 = 9800 nM T79062 CT9L0D 3084440 Ki = 80 nM T79062 C6SA2G 3132842 Ki = 37200 nM T79062 CNX8I1 3245407 IC50 > 1000 nM T79062 CX8W7I 3377940 Ki = 1700 nM T79062 CS8KE2 3649661 Ki = 472 nM T79062 C6SHA4 4713248 Ki = 950 nM T79062 CRUB15 4723431 Ki = 1281 nM T79062 C7PX9E 4790508 Ki = 197 nM T79062 C9NKP1 5216959 Ki = 265 nM T79062 C4BKS2 5242341 Ki = 502 nM T79062 C4J3HP 5640104 Ki = 3490 nM T79062 CGM63Y 6540428 Ki = 12.59 nM T79062 C0QCK1 6918455 Ki = 3981.07 nM T79062 CW0ZE5 6918542 Ki = 600 nM T79062 CC5PQ0 6918601 Ki > 5800 nM T79062 C1WXY3 6918603 Ki < 7943.28 nM T79062 CD0Z4I 6918648 Ki = 3162.28 nM T79062 C8AL9V 6918689 Ki < 100000 nM T79062 CI0X2F 7059581 Ki = 1 nM T79062 C2F3BY 7125890 Ki = 9566 nM T79062 CUD06Z 9796627 Ki = 1600 nM T79062 CFC9Y5 9799318 Ki = 6.457 nM T79062 CG0UK3 9803482 Ki = 16.98 nM T79062 CE0DI5 9804612 Ki = 79.43 nM T79062 CNX4F0 9805456 Ki < 5011.87 nM T79062 CWOS30 9817810 Ki = 29 nM T79062 CFBH76 9820952 Ki = 31.62 nM T79062 CBN06W 9839050 Ki = 13 nM T79062 CE3W4V 9845006 Ki = 2.138 nM T79062 CM13ZV 9856041 Ki = 24000 nM T79062 C0ZR3E 9861687 IC50 > 1000 nM T79062 CNCK78 9862256 Ki = 460 nM T79062 C4H7DK 9864569 IC50 < 50 nM T79062 CB1F0C 9867475 Ki = 1300 nM T79062 C7AB8O 9870053 Ki < 5011.87 nM T79062 CQ4LC2 9872676 Ki = 1750 nM T79062 CCLN49 9878197 Ki = 49 nM T79062 C9NF3D 9881600 Ki = 0.6 nM T79062 C08DBF 9885982 Ki = 3 nM T79062 CL1W0B 9887186 Ki = 5.754 nM T79062 CJW1P5 9888494 Ki = 2.239 nM T79062 C6N8UE 9889681 Ki < 10000 nM T79062 CM52WU 9890119 Ki = 2511.89 nM T79062 CEG1K5 9891002 Ki = 1584.89 nM T79062 C7QMK5 9891617 Ki < 5011.87 nM T79062 CEL29O 9891618 Ki = 1995.26 nM T79062 C3J8GU 9892409 Ki < 7943.28 nM T79062 CAM25C 9894665 Ki = 10 nM T79062 CUN81Q 9905249 Ki > 10000 nM T79062 CYWQ50 9906447 Ki > 10000 nM T79062 C9B3EA 9911844 Ki = 7.24 nM T79062 C78MDV 9913554 Ki = 1000 nM T79062 CR9KM0 9921064 Ki = 290 nM T79062 C4UYZ7 9927441 Ki = 3700 nM T79062 CYVZ47 9934284 Ki = 39.81 nM T79062 CO2RS8 9934709 Ki = 0.6761 nM T79062 CWO45F 9935387 Ki = 630.96 nM T79062 CX6E8C 9945703 Ki = 6 nM T79062 CQ04ZS 9950396 Ki = 400 nM T79062 CK8NR2 9954121 Ki < 10000 nM T79062 CHOJ30 9956365 Ki = 3.548 nM T79062 CFR41N 9957068 Ki < 3981.07 nM T79062 CFN50J 9978683 Ki = 579 nM T79062 CS40QN 10015688 Ki = 0.7 nM T79062 CV7R9F 10020040 Ki = 335.9 nM T79062 CK18LT 10020895 Ki > 5000 nM T79062 C2EUY0 10035109 Ki > 10000 nM T79062 C57TZR 10042333 Ki = 1345 nM T79062 C0KWB6 10062885 Ki = 1.1 nM T79062 CR68SH 10064053 Ki = 9.78 nM T79062 C8Z6MA 10067306 IC50 = 1217 nM T79062 CKA5F4 10084076 Ki = 18 nM T79062 C93RNG 10090247 Ki = 7 nM T79062 CA5H7K 10106205 Ki = 16 nM T79062 C4Q3UL 10154897 Ki = 3 nM T79062 C7F1ED 10183148 IC50 = 135000 nM T79062 CW09SL 10202089 Ki = 6 nM T79062 C4Q2SH 10249573 Ki = 10 nM T79062 CMRA02 10257042 Ki < 794.33 nM T79062 CH31DX 10267394 Ki = 412.3 nM T79062 CTWJ70 10274894 Ki = 2.042 nM T79062 CU89JD 10314060 Ki = 102.8 nM T79062 C9IAV3 10346043 Ki = 1.023 nM T79062 CA7IM5 10379532 Ki = 1.096 nM T79062 CR3KU9 10380133 IC50 > 5000 nM T79062 CMZA83 10383646 Ki = 753 nM T79062 C4L5PQ 10404657 Ki = 8.511 nM T79062 C04WGF 10407367 IC50 = 511 nM T79062 C4TPN1 10413595 Ki = 0.3162 nM T79062 C2B0IU 10421236 IC50 > 10000 nM T79062 CR4LS0 10430623 Ki = 1563 nM T79062 CD7U5I 10433930 Ki = 1.995 nM T79062 CO7IV6 10450593 Ki = 0.1995 nM T79062 COV85C 10472143 Ki = 14 nM T79062 C5LBS7 10472158 IC50 = 1362 nM T79062 C26KCR 10475231 Ki = 2 nM T79062 CEF2O6 10478367 Ki = 1412 nM T79062 CL70NJ 10499156 Ki = 10 nM T79062 CN29IF 10500557 Ki = 2.138 nM T79062 CWH7R8 10521887 Ki = 26.33 nM T79062 C9B7LR 10552788 Ki = 19.95 nM T79062 CHE80N 10573876 Ki = 1.995 nM T79062 CAVR62 10596321 Ki = 10 nM T79062 CO23YX 10597140 Ki = 15.85 nM T79062 CZ6WS8 10619437 Ki = 125.89 nM T79062 CAPO49 10638372 Ki = 105 nM T79062 CK08CW 10643153 Ki = 10000 nM T79062 CN40TJ 10668422 Ki < 1000 nM T79062 CBE87R 10706626 Ki = 13.4 nM T79062 CU32PG 10714877 Ki = 10.35 nM T79062 C1PG3A 10715573 Ki = 31.62 nM T79062 CJ4HC8 10715998 Ki = 15.85 nM T79062 CZ3A0O 10737314 Ki = 100 nM T79062 CIVN21 10767321 Ki = 15.85 nM T79062 C2AFT6 10785644 Ki = 1584.89 nM T79062 C3SWV9 10785714 Ki = 5 nM T79062 C75SKC 10811746 Ki = 3.802 nM T79062 CG4X1R 10834268 Ki = 1.862 nM T79062 C8MHZ9 10835110 Ki = 3.981 nM T79062 C5Q4IJ 10862697 Ki = 2.344 nM T79062 CFY4V1 10862787 Ki = 12 nM T79062 CVT7J1 10873805 Ki = 7.32 nM T79062 CNEP25 10884517 Ki = 7.943 nM T79062 C67UIY 10884717 Ki = 6.457 nM T79062 CRI50E 10885636 IC50 = 1440 nM T79062 C9C2FI 10895284 Ki = 72.44 nM T79062 CD4YL2 10896196 Ki = 19.05 nM T79062 CX65PW 10907460 IC50 = 2040 nM T79062 CEGJ41 10917174 Ki = 6.026 nM T79062 CU09AV 10937901 IC50 = 762 nM T79062 C7PWT9 10938620 Ki = 109.65 nM T79062 CA42MT 10939416 Ki = 8.71 nM T79062 CNB39C 10947658 Ki = 12 nM T79062 CSLT97 10949380 IC50 = 663 nM T79062 C2MBP7 10949445 Ki = 8.128 nM T79062 C74SOA 10950559 Ki = 74 nM T79062 C47MYE 10960943 Ki = 97.72 nM T79062 CJD58C 10971401 Ki = 4.786 nM T79062 C51NOQ 10982183 Ki < 10000 nM T79062 CK6VF7 10991109 Ki = 63 nM T79062 C4O7MD 10994400 Ki = 101 nM T79062 CJC9K4 11005810 IC50 = 998 nM T79062 C3FIP5 11016205 Ki = 3.68 nM T79062 CS0Z2D 11024311 Ki < 10000 nM T79062 CRS62E 11025847 Ki = 3.548 nM T79062 C0HA7O 11047374 Ki = 1.995 nM T79062 C23JHR 11047568 IC50 = 1430 nM T79062 C80UIZ 11048252 Ki = 416.87 nM T79062 CONV96 11058267 Ki = 45.71 nM T79062 CD4BW6 11058564 Ki = 43.65 nM T79062 CZN25U 11059148 Ki = 23.99 nM T79062 CG41BK 11071079 IC50 = 726 nM T79062 C15USQ 11101733 Ki = 19.05 nM T79062 C7OFQ4 11102049 Ki = 29.51 nM T79062 CCJ1U3 11112531 Ki = 147 nM T79062 C7DE0U 11113605 IC50 = 1170 nM T79062 CVE8T3 11121216 Ki = 31 nM T79062 C5I0XL 11133795 Ki = 223.87 nM T79062 C0VZK2 11143387 Ki = 9.7 nM T79062 CS90QD 11145126 Ki = 7.079 nM T79062 CYJ79P 11153905 Ki = 2.55 nM T79062 C8ZN3B 11166042 Ki = 37 nM T79062 CEHV65 11173572 Ki = 13.4 nM T79062 C6CL1Y 11178830 Ki = 125.89 nM T79062 C0W4SM 11186523 Ki = 6.5 nM T79062 CXQ3K0 11186985 Ki = 2.91 nM T79062 C5J4NR 11199511 Ki = 8 nM T79062 C9N5QU 11200511 Ki = 74 nM T79062 C90WSG 11248705 Ki = 125.89 nM T79062 CM08DU 11259115 Ki = 200 nM T79062 C4S2VF 11277147 Ki = 17.6 nM T79062 CY6MX5 11282296 EC50 = 2460 nM T79062 CW40XM 11294248 Ki = 251 nM T79062 C9BLC7 11304596 Ki = 501.19 nM T79062 CJS9C0 11304851 IC50 = 25000 nM T79062 CI79LV 11307899 Ki = 6.31 nM T79062 C1VSE5 11327643 Ki = 1000 nM T79062 CGD42N 11361090 Ki > 5000 nM T79062 CXW6B5 11373831 Ki = 19 nM T79062 CBV52J 11384146 Ki = 24 nM T79062 C1BP0U 11385380 Ki > 1000 nM T79062 CF4OX6 11397149 Ki = 79.43 nM T79062 C30ZMW 11397459 Ki = 200 nM T79062 C7GXP9 11397799 Ki = 9 nM T79062 C85LYP 11430418 IC50 = 1000 nM T79062 CNF28A 11432177 EC50 = 6320 nM T79062 CJK2S4 11453751 Ki = 221 nM T79062 CMFC18 11453756 Ki = 200 nM T79062 C9K8UW 11515799 Ki = 7.65 nM T79062 CVAC51 11524003 Ki = 1.19 nM T79062 C7YRP3 11524413 Ki = 0.38 nM T79062 CFW50Y 11525867 Ki = 9.5 nM T79062 C2M0JG 11532105 Ki = 40 nM T79062 C5VHK0 11536843 Ki = 5.1 nM T79062 C0YZ7L 11536844 Ki = 3.3 nM T79062 C1V5CH 11559090 Ki > 10000 nM T79062 C14HEP 11560285 Ki = 296 nM T79062 C1HP5K 11566558 Ki = 4.31 nM T79062 CNH1K4 11568826 Ki = 520 nM T79062 C8NMI4 11575479 Ki = 600 nM T79062 C1I4DF 11582132 Ki = 25 nM T79062 C6D1MA 11584660 Ki > 1995.26 nM T79062 C1M2CP 11589069 Ki = 0.38 nM T79062 CU45DK 11595209 Ki > 10000 nM T79062 CE9W6J 11595790 Ki = 16.8 nM T79062 CGX8F6 11596869 Ki > 3980000 nM T79062 CX5ZM0 11603891 Ki = 5.38 nM T79062 C8EPV2 11610908 Ki = 64 nM T79062 CUA05E 11617668 Ki = 5.4 nM T79062 CD4HR8 11633354 Ki = 2.1 nM T79062 C2OU7Y 11638332 Ki > 10000 nM T79062 C9OLN0 11646336 Ki = 5 nM T79062 CJBV31 11652871 IC50 = 118100 nM T79062 CCX0S1 11653869 Ki = 0.49 nM T79062 CO1L8J 11661471 Ki = 1.02 nM T79062 C4L7TV 11662592 Ki = 4.48 nM T79062 CD91CP 11666595 Ki = 33 nM T79062 CXRC27 11667458 Ki = 10.9 nM T79062 C42RHW 11674602 Ki = 94 nM T79062 CL31JB 11683077 Ki = 11.1 nM T79062 CEQ6W7 11694810 Ki = 4.3 nM T79062 C2QCF5 11697434 Ki = 18 nM T79062 CHR8U4 11697659 Ki = 2.81 nM T79062 C3IML2 11709509 Ki = 0.3 nM T79062 C1N7MO 11725453 Ki = 1 nM T79062 CV82QX 11729084 Ki = 25.12 nM T79062 CLYJ75 11729823 Ki = 8.76 nM T79062 C7PVL8 11730467 IC50 = 2130 nM T79062 CG72CS 11732538 Ki = 20 nM T79062 CMO0I9 11739679 Ki = 1555 nM T79062 C57IKL 11740526 Ki = 9.772 nM T79062 CPG15O 11743399 IC50 > 1000 nM T79062 CYV02C 11747350 Ki = 510 nM T79062 C3F5DX 11761059 IC50 = 4420 nM T79062 C9LUA7 11773414 Ki = 800 nM T79062 C37LEP 11785183 EC50 = 1820 nM T79062 C7A2QD 11793826 Ki = 630.96 nM T79062 C3PY7W 11811833 Ki = 21.88 nM T79062 CQV92N 11825614 Ki = 10.47 nM T79062 CW4BC2 11826723 Ki = 12.3 nM T79062 CXLW54 11948707 Ki = 328 nM T79062 C8JQL7 11957735 IC50 = 1713 nM T79062 C1QY2P 12005903 Ki = 15770 nM T79062 C8EDN0 12088080 Ki = 3 nM T79062 C8RB6W 12088082 Ki = 9 nM T79062 CLC82F 12374770 Ki = 176 nM T79062 CCG14E 13091356 Ki = 420 nM T79062 CYN95Z 13091359 Ki = 97 nM T79062 C4V6AS 14135325 IC50 = 179000 nM T79062 CAO70J 14748689 IC50 = 949 nM T79062 C7VAI1 15011772 IC50 > 10000 nM T79062 C30CHU 15512229 Ki < 316.23 nM T79062 CKBD37 15542627 Ki = 17.38 nM T79062 C65SCN 15599151 Ki = 1240 nM T79062 CTPX97 15803947 Ki = 1.3 nM T79062 C1LWZ6 16006605 Ki = 2.4 nM T79062 CK36NS 16006607 Ki = 1 nM T79062 C3M8GJ 16026344 Ki = 5232 nM T79062 C1SR0O 16071847 Ki > 5000 nM T79062 CD3E8L 16093484 Ki = 8.7 nM T79062 CEW91O 16093485 Ki = 2.5 nM T79062 CZ1WJ4 16117151 Ki = 3970 nM T79062 CM32ZX 16117153 Ki > 5000 nM T79062 CXTB90 16117279 Ki = 3216 nM T79062 C1F2LS 16118795 Ki > 5000 nM T79062 C69VDS 16118923 Ki > 5000 nM T79062 CZ2IS9 16660294 Ki > 10000 nM T79062 CT9GP4 16763549 Ki = 13100 nM T79062 CR63LE 17055181 Ki = 3700 nM T79062 C0QX5J 17374371 Ki = 12590 nM T79062 CB2J3R 17747575 IC50 > 100 nM T79062 C42YEX 18133517 Ki = 3187 nM T79062 CI90UP 18133518 Ki = 2544 nM T79062 C7R1IG 18137015 Ki = 1029 nM T79062 C4I1FW 18137017 Ki = 1342 nM T79062 C07EOI 18137020 Ki = 1417 nM T79062 C9PV8A 18180076 IC50 = 1582 nM T79062 CI6TS8 18377342 Ki = 562.34 nM T79062 CHFJ09 18377388 Ki = 173.78 nM T79062 C5KB2J 18377409 Ki = 15.85 nM T79062 CI91VX 18377415 Ki = 812.83 nM T79062 CXR67I 18663036 Ki = 18.4 nM T79062 C6AOE8 19426635 IC50 = 18.62 nM T79062 CUI3R1 19605739 Ki = 1 nM T79062 C7T8JC 19958494 Ki = 318.2 nM T79062 C6LI5E 19958507 Ki = 411 nM T79062 CBY03N 20846175 Ki < 10000 nM T79062 CISE25 21091965 Ki = 80 nM T79062 C6H9WC 21092408 Ki = 88 nM T79062 C3T5HF 21509921 Ki = 100 nM T79062 CFN81Q 21527771 Ki = 656 nM T79062 CH59WN 21533446 Ki = 1044 nM T79062 C4B0TN 21557475 Ki = 1200 nM T79062 CT7XG9 21830793 Ki = 12.9 nM T79062 C9X8PI 22001618 Ki = 2.6 nM T79062 CBN84K 22065997 Ki = 212.9 nM T79062 C1QBE0 22273749 Ki = 11.22 nM T79062 C6UXL4 22330705 Ki = 21400 nM T79062 CZG9S2 22425072 Ki = 12710 nM T79062 CW0V5M 22449331 Ki = 4.467 nM T79062 CPD8Q7 22549784 Ki = 26650 nM T79062 CZ7J4B 22857296 Ki = 6.4 nM T79062 C0L5QK 23111951 Ki = 270 nM T79062 CY10BQ 23133427 Ki = 2.7 nM T79062 C5BUL7 23151712 Ki = 43 nM T79062 C3IF7P 23151734 Ki = 185 nM T79062 C0NI3J 23290944 Ki = 198 nM T79062 C57MVP 23369416 Ki = 3.4 nM T79062 C6HE8J 23369421 Ki = 26 nM T79062 CAE7K1 23369450 Ki = 1838 nM T79062 CWQ2X3 23369455 Ki = 48 nM T79062 C7EPU0 23369457 Ki = 1029 nM T79062 CRT2Z3 23661667 Ki = 54 nM T79062 CHGE36 23661734 Ki = 46 nM T79062 C5ZSR7 23661735 Ki = 1200 nM T79062 CQE1N7 23906630 Ki = 16020 nM T79062 CD7CV6 24771120 Ki = 6900 nM T79062 CCEH06 24781896 IC50 > 100 nM T79062 CD86PT 24781897 IC50 > 100 nM T79062 CP7TJ3 24781898 IC50 > 100 nM T79062 CF17PW 24781899 IC50 > 100 nM T79062 C1JSY8 24781900 IC50 > 100 nM T79062 CJI2O1 24782049 IC50 > 100 nM T79062 CK9T1F 24782050 IC50 > 100 nM T79062 C2O7MV 24782051 IC50 > 100 nM T79062 C0G3RV 24782052 IC50 > 100 nM T79062 CR8DV4 24782058 IC50 > 100 nM T79062 C58AMS 24829343 Ki = 0.79 nM T79062 CDC91N 24839550 Ki < 10000 nM T79062 CY21RE 24841480 Ki = 330 nM T79062 CT2YG6 24853955 Ki = 0.6 nM T79062 C2KD1T 24854037 Ki = 0.66 nM T79062 C1BPD9 24854039 Ki = 5.3 nM T79062 CGPC24 24854040 Ki = 8.27 nM T79062 CM01LB 24854041 Ki = 0.67 nM T79062 CI7G6M 24854043 Ki = 4.75 nM T79062 C4WUP5 24854044 Ki = 1.1 nM T79062 CY1XA8 24854103 Ki = 6.99 nM T79062 C42KBQ 24854105 Ki = 1.96 nM T79062 CUW23K 24854106 Ki = 44 nM T79062 CX7MK6 24854108 Ki = 33.38 nM T79062 CS90OD 24854109 Ki = 21 nM T79062 CFHM49 24854111 Ki = 1.45 nM T79062 C80ANM 24854181 Ki = 1.24 nM T79062 CSL8E3 24854183 Ki = 1.5 nM T79062 CFR74S 24854185 Ki = 1.8 nM T79062 CW2Z5A 24854186 Ki = 25.4 nM T79062 C9GYO8 24854187 Ki = 0.43 nM T79062 CB9M0N 24854266 Ki = 9.07 nM T79062 C0LQ1R 24854267 Ki = 3.4 nM T79062 CP23KC 24854269 Ki = 6.57 nM T79062 CI5LC8 24854270 Ki = 9.46 nM T79062 CCUS10 24854272 Ki = 5.97 nM T79062 CFX96I 24854273 Ki = 0.4 nM T79062 C6Y3AG 24854368 Ki = 2.07 nM T79062 CTS4E5 24854369 Ki = 2.55 nM T79062 COZ84H 24854370 Ki = 5.11 nM T79062 C3X9MD 24854371 Ki = 0.6 nM T79062 C7ZEF0 24856058 IC50 > 10000 nM T79062 C3HK0J 24865725 Ki = 19.95 nM T79062 C0O6FX 24865727 Ki = 15.85 nM T79062 C98ZIV 24882509 IC50 = 11.99 nM T79062 C6L7KS 24887518 Ki < 3162.28 nM T79062 CAOF91 24894071 IC50 > 10000 nM T79062 CMN75S 24901425 Ki = 1659.59 nM T79062 CF7IV1 24963856 Ki = 6.2 nM T79062 C8DJG7 24963860 Ki = 8.6 nM T79062 C35XOJ 24964217 Ki = 8.4 nM T79062 CP6K8J 25024727 IC50 > 10000 nM T79062 CI95EF 25192947 Ki = 0.47 nM T79062 CKAS93 25256850 Ki = 6 nM T79062 CW07GN 25256855 Ki = 7 nM T79062 CM2T9Y 25263297 Ki = 5100 nM T79062 CFJM71 25263302 Ki = 5800 nM T79062 CHJ35A 32354149 Ki = 885 nM T79062 CS5QG1 35391328 Ki = 773 nM T79062 C8G7EY 36418162 IC50 = 476 nM T79062 CDV36I 37219401 Ki = 855 nM T79062 CG56DF 42388639 IC50 = 20 nM T79062 C6VL8I 42388965 IC50 = 140 nM T79062 CS2G3E 42388975 IC50 = 289 nM T79062 CJ8FH4 42389129 IC50 = 681 nM T79062 CO51RQ 42389139 IC50 > 10000 nM T79062 CBV62E 42389293 IC50 = 3241 nM T79062 CNV94Z 42389303 IC50 = 9314 nM T79062 CSRX20 42389457 IC50 = 53 nM T79062 CH5QX6 42389467 IC50 = 47 nM T79062 CV9C4D 42428409 Ki = 78 nM T79062 C1SD3E 42618253 Ki = 1230 nM T79062 C0BWG1 42618254 Ki = 902 nM T79062 CAG71H 42618255 Ki = 864 nM T79062 CQ96KL 42618256 Ki = 566 nM T79062 CC1Z7P 42618257 Ki = 1867 nM T79062 CFB70T 42618258 Ki = 17960 nM T79062 CJV5N3 42618259 Ki = 2500 nM T79062 CHA26S 42618260 Ki = 296 nM T79062 CX1KC4 42618261 Ki = 168 nM T79062 C2VWK7 42618262 Ki = 267 nM T79062 CV0CD8 42618263 Ki = 243 nM T79062 CS5TJ8 42618264 Ki = 38 nM T79062 CKOJ59 42618265 Ki = 20 nM T79062 C4J9RQ 42618266 Ki = 78 nM T79062 C16TUL 42618267 Ki = 11 nM T79062 CH3NO7 42618269 Ki = 21 nM T79062 CMGJ03 42618270 Ki = 134 nM T79062 CR6OX0 42618271 Ki > 5000 nM T79062 C7SN5E 42618272 Ki = 31 nM T79062 C3VR7E 42618273 Ki = 335 nM T79062 CA0B9F 42625181 Ki = 68 nM T79062 C3L0TN 42625183 Ki = 69 nM T79062 CW0OU4 42625185 Ki > 1000 nM T79062 CHY12B 42625186 Ki > 1000 nM T79062 CP5X3K 42625188 Ki > 1000 nM T79062 C8QSX3 42625267 Ki = 193 nM T79062 CTM69J 42625269 Ki = 350 nM T79062 CPDG98 42625353 Ki = 63 nM T79062 CK3QD2 42625354 Ki > 1000 nM T79062 CJ64FG 42625356 Ki = 250 nM T79062 C27KEF 42625359 Ki = 160 nM T79062 CN81SE 42625440 Ki = 7 nM T79062 CF7DM0 42625445 Ki = 22 nM T79062 CJI51X 42625446 Ki = 69 nM T79062 CLH7Y0 42626289 Ki = 158 nM T79062 C75QPL 42626291 Ki = 203 nM T79062 C5VTZ6 42626293 Ki = 74 nM T79062 C70SWL 42626361 Ki = 63 nM T79062 CY7W2J 42631003 Ki = 0.153 nM T79062 CV2X5B 42635027 IC50 = 89 nM T79062 CBSD79 42635028 IC50 = 384 nM T79062 CR1S3J 42635029 IC50 = 339 nM T79062 CS9Q3H 42635204 IC50 = 12 nM T79062 C5XBV7 42635205 IC50 = 567 nM T79062 CQ2M5S 42635387 IC50 = 124 nM T79062 CR3KM7 42635388 IC50 = 107 nM T79062 C8TFQ9 42635389 IC50 = 580 nM T79062 CFO4Y1 42635570 IC50 = 223 nM T79062 CWU54L 42635571 IC50 = 373 nM T79062 CV27CE 42635572 IC50 = 377 nM T79062 CJ3NP5 42636941 IC50 > 1000 nM T79062 C0AI7N 43229249 Ki = 354.81 nM T79062 C2RSL9 43840296 Ki = 226 nM T79062 CJ41QV 44126269 Ki = 0.389 nM T79062 CVG6X1 44209472 Ki = 208 nM T79062 CD5AB7 44209480 Ki = 90 nM T79062 C2FDB1 44250364 IC50 > 10000 nM T79062 C8MC0Q 44251387 IC50 > 10000 nM T79062 C5YEA8 44251388 IC50 > 10000 nM T79062 C0BSF6 44251389 IC50 > 10000 nM T79062 CP8S2J 44266156 Ki = 4.467 nM T79062 CM0CW8 44266160 Ki = 6.918 nM T79062 C0P8IF 44266163 Ki = 0.4074 nM T79062 CU67NF 44266164 Ki = 9.333 nM T79062 C14ACY 44266178 Ki = 37.15 nM T79062 CN3ES2 44266182 Ki = 2.042 nM T79062 CKLS45 44266203 Ki = 14.13 nM T79062 CARU58 44266221 Ki = 0.5623 nM T79062 CA1WJ4 44266222 Ki = 2.754 nM T79062 CS2MU8 44266229 Ki = 20.42 nM T79062 CZ84XC 44266244 Ki = 9.12 nM T79062 CR16DY 44266245 Ki = 11.75 nM T79062 CVHM20 44266253 Ki = 27.54 nM T79062 CK7AF0 44266267 Ki = 25.12 nM T79062 C1FTY0 44266268 Ki = 1.66 nM T79062 CU61ZS 44266284 Ki = 11.22 nM T79062 C0C6RL 44266289 Ki = 10.23 nM T79062 C5NS9O 44266315 Ki = 2.512 nM T79062 CO5H2Q 44266317 Ki = 18.62 nM T79062 C6OW2N 44268087 Ki = 32 nM T79062 CNHE76 44276598 Ki = 2.138 nM T79062 CC2OD4 44278111 Ki > 10000 nM T79062 CRMA84 44278114 Ki = 713 nM T79062 CF0Y4M 44278115 Ki > 10000 nM T79062 CA93MC 44319240 Ki = 12.59 nM T79062 C34FTE 44319435 Ki = 8.318 nM T79062 CW16JD 44324737 Ki > 1000 nM T79062 CA84SN 44324765 Ki > 1000 nM T79062 COA3H4 44324800 Ki > 1000 nM T79062 CY04JW 44324972 Ki > 1000 nM T79062 C5VLY2 44326733 Ki = 9 nM T79062 CT7DN4 44327688 Ki = 2.399 nM T79062 CER86D 44327952 Ki = 83 nM T79062 CP9B2K 44340834 Ki = 1.82 nM T79062 CB23YQ 44340835 Ki = 0.7943 nM T79062 CC25ZK 44340836 Ki = 0.5012 nM T79062 CZBQ72 44340850 Ki = 0.8318 nM T79062 CTM65V 44340854 Ki = 0.7079 nM T79062 C6F9XL 44340882 Ki = 57.54 nM T79062 C2S1ZT 44340883 Ki = 6.457 nM T79062 CG6PD8 44340897 Ki = 22.91 nM T79062 CQ3WH6 44341114 Ki = 6.31 nM T79062 C9BDG2 44341126 Ki = 6.457 nM T79062 CK37NE 44341130 Ki = 25.7 nM T79062 CO0ZY5 44341131 Ki = 165.96 nM T79062 CD9ZS8 44342270 IC50 = 849 nM T79062 CPWJ26 44343212 Ki = 39.81 nM T79062 CMX45U 44348383 IC50 = 2.2 nM T79062 CUXH48 44352308 Ki = 1460 nM T79062 C3LKN1 44364048 Ki = 3.162 nM T79062 CND4W7 44368304 Ki = 19.95 nM T79062 C6CUM2 44368306 Ki = 31.62 nM T79062 CH3G4F 44368358 Ki = 31.62 nM T79062 C2S8AQ 44368373 Ki = 100000 nM T79062 C1EO8C 44368383 Ki = 1584.89 nM T79062 CAEZ93 44368384 Ki = 630.96 nM T79062 CK9OQ3 44368683 Ki = 125.89 nM T79062 CB0E1J 44368705 Ki = 10 nM T79062 CS21UK 44368731 Ki = 1.995 nM T79062 CRF67K 44368732 Ki = 3.981 nM T79062 C61PEQ 44368754 Ki = 15.85 nM T79062 CT2BR5 44372581 Ki = 5.012 nM T79062 C08EKS 44374206 Ki = 1200 nM T79062 CVL3U2 44374207 Ki = 7.2 nM T79062 CV8CP3 44374225 Ki = 22 nM T79062 C7FE5A 44374226 Ki = 6800 nM T79062 CX9S1K 44374227 Ki = 3200 nM T79062 C04WKH 44374233 Ki = 4.1 nM T79062 CB2S7T 44374234 Ki = 100 nM T79062 CV62ZP 44374298 Ki = 170 nM T79062 CJ4A2U 44374299 Ki = 12 nM T79062 C4VXQ1 44388858 Ki = 4.3 nM T79062 CTPG47 44388956 Ki > 2000 nM T79062 C1UMV6 44393001 Ki = 60 nM T79062 C64IKJ 44393004 Ki = 4 nM T79062 CT8Y5A 44393007 Ki = 4 nM T79062 C1F5IX 44393021 Ki = 13 nM T79062 C9VH1B 44393022 Ki = 16 nM T79062 CG9S1O 44393045 Ki = 2 nM T79062 CGRD59 44393052 Ki = 23 nM T79062 CBJ84O 44393053 Ki = 54 nM T79062 CPS9T7 44393056 Ki > 1000 nM T79062 C4HVE3 44393057 Ki > 1000 nM T79062 CKV3Z0 44393069 Ki = 3 nM T79062 C7HIJ9 44393072 Ki = 10 nM T79062 C20PMS 44393073 Ki = 0.4 nM T79062 C1E0QH 44393074 Ki = 36 nM T79062 C3H6ML 44393075 Ki = 8 nM T79062 C53UVJ 44393088 Ki = 2 nM T79062 C89NKB 44393089 Ki > 1000 nM T79062 C2QX0I 44393090 Ki > 1000 nM T79062 C0F9MP 44393091 Ki = 0.3 nM T79062 CCS5Q4 44393092 Ki = 0.4 nM T79062 C1KBZ7 44393093 Ki > 1000 nM T79062 CO6EY0 44393113 Ki = 2 nM T79062 C9GEU3 44393114 Ki = 33 nM T79062 CX4C9P 44393133 Ki = 6 nM T79062 CE03ZW 44393134 Ki = 1 nM T79062 C69CFB 44393154 Ki > 41000 nM T79062 CP9K0J 44393161 Ki = 2 nM T79062 CY60BQ 44393162 Ki > 1000 nM T79062 CG5UE1 44393169 Ki = 0.3 nM T79062 CG18AU 44393170 Ki = 5 nM T79062 CZ18RL 44393171 Ki = 5 nM T79062 CHV6D3 44393180 Ki = 0.6 nM T79062 CZB65R 44393192 Ki = 0.4 nM T79062 CK85EB 44393193 Ki = 0.4 nM T79062 CVC86L 44393228 Ki = 3 nM T79062 C7AR1C 44393229 Ki = 4 nM T79062 C4B0OI 44397588 Ki = 1000 nM T79062 C5FP0R 44397589 Ki = 1258.93 nM T79062 CE3G8U 44397670 Ki = 3981.07 nM T79062 CX7O9S 44401041 Ki = 80 nM T79062 C5XC2B 44401042 Ki = 92 nM T79062 CD56EA 44401105 Ki = 35 nM T79062 CW3PC2 44401106 Ki = 34 nM T79062 C9WH7P 44401164 Ki = 6.2 nM T79062 C9CWX1 44401194 Ki = 57 nM T79062 CXT84G 44401243 Ki = 251 nM T79062 C1B4QL 44403095 Ki > 10000 nM T79062 C1YL7Z 44403098 Ki > 10000 nM T79062 CFV98A 44403101 Ki > 10000 nM T79062 C6OY9S 44403102 Ki > 10000 nM T79062 CH4SX6 44403105 Ki > 10000 nM T79062 C4LKC1 44404394 Ki = 342 nM T79062 C3EJ4G 44404396 Ki > 10000 nM T79062 CG87PW 44409290 Ki > 1000 nM T79062 CXO64D 44437860 Ki = 107 nM T79062 CWO35N 44437861 Ki > 5000 nM T79062 CKZF16 44439165 Ki = 39.81 nM T79062 CA4HZ3 44439167 Ki = 79.43 nM T79062 CRC2Y5 44439387 Ki = 800 nM T79062 C3ZT7I 44439388 Ki = 3500 nM T79062 CKU9N8 44439389 Ki = 7800 nM T79062 C20VDP 44439390 Ki = 45 nM T79062 C6RKA9 44439391 Ki = 36 nM T79062 CI9D7G 44439392 Ki = 20 nM T79062 CDE27X 44439393 Ki = 35 nM T79062 CIQW67 44439394 Ki = 170 nM T79062 CV93LJ 44439395 Ki = 46 nM T79062 CPX5Q2 44439396 Ki = 200 nM T79062 C2R0SX 44439397 Ki = 2200 nM T79062 C4CMV7 44439398 Ki = 400 nM T79062 C8YQ4P 44439399 Ki = 500 nM T79062 C6YA9O 44439400 Ki = 5300 nM T79062 C89ZPX 44439401 Ki = 25000 nM T79062 CE60JL 44439402 Ki = 2700 nM T79062 C65GSE 44439403 Ki = 1000 nM T79062 CKUG90 44439404 Ki = 100 nM T79062 CTYP87 44439405 Ki = 300 nM T79062 C3UBA6 44439406 Ki > 300000 nM T79062 C7HV8X 44439407 Ki = 36000 nM T79062 CD4T3S 44439408 Ki = 200 nM T79062 C07XPE 44439409 Ki = 100 nM T79062 CMU43Q 44439410 Ki = 3600 nM T79062 C2S6HQ 44448054 Ki = 55 nM T79062 C3Z7FI 44451927 IC50 = 119.95 nM T79062 CSD7R5 44451929 IC50 = 2197.86 nM T79062 C3MCY7 44451930 IC50 = 1300 nM T79062 C3R7BH 44451931 IC50 = 369.83 nM T79062 CRFN53 44451952 IC50 = 260.02 nM T79062 CZE3T1 44451953 IC50 = 199.99 nM T79062 CJTX92 44451954 IC50 = 190 nM T79062 CINR86 44451957 IC50 = 2500 nM T79062 CK4GN8 44451959 IC50 = 500 nM T79062 CL29TJ 44451979 IC50 = 620 nM T79062 C57SBC 44451980 IC50 = 16 nM T79062 CEST18 44451982 IC50 = 54.95 nM T79062 CV7EY2 44451984 IC50 = 500 nM T79062 C7L9DK 44451985 IC50 = 939.72 nM T79062 C15JOU 44451986 IC50 = 510 nM T79062 CM34IO 44452005 IC50 = 190 nM T79062 C39KGW 44452006 IC50 = 269.77 nM T79062 CRN4F8 44452007 IC50 = 49 nM T79062 CY43VF 44452008 IC50 = 42 nM T79062 CW80FP 44452010 IC50 = 680 nM T79062 C3L6IQ 44452037 IC50 = 28.97 nM T79062 CR4N5K 44452038 IC50 = 1199.5 nM T79062 CN6PT7 44452039 IC50 = 130.02 nM T79062 CB0CK5 44452040 IC50 = 769.13 nM T79062 C74KEA 44452041 IC50 = 769.13 nM T79062 CL2EH4 44452042 IC50 = 8994.98 nM T79062 CO1W6H 44452078 IC50 = 97 nM T79062 CT2VN0 44452080 IC50 = 199.99 nM T79062 CA91RH 44452081 IC50 = 419.76 nM T79062 C6U4YS 44452082 IC50 = 928.97 nM T79062 C7DAM2 44452084 IC50 > 10000 nM T79062 CP1E6V 44452114 IC50 = 1000 nM T79062 COR7N6 44452115 IC50 = 16 nM T79062 C65HFP 44452117 IC50 = 470 nM T79062 C8F7IQ 44452118 IC50 = 349.95 nM T79062 CN4YL1 44452139 IC50 = 230 nM T79062 CMP20V 44452141 IC50 = 680 nM T79062 CG1C6X 44452142 IC50 = 92 nM T79062 C7A9JI 44452143 IC50 = 26 nM T79062 C78UTQ 44452144 IC50 = 1999.86 nM T79062 CQR12V 44452145 IC50 > 10000 nM T79062 CF3H6V 44452166 IC50 = 19 nM T79062 C6SC1Q 44452167 IC50 = 91 nM T79062 C56JMP 44452169 IC50 > 10000 nM T79062 CQ5U1I 44452170 IC50 = 20.99 nM T79062 CX8OK7 44452171 IC50 = 45 nM T79062 CS72NU 44452193 IC50 = 54.95 nM T79062 C5ZF1H 44452195 IC50 = 97.95 nM T79062 CTAP34 44452196 IC50 = 199.99 nM T79062 CUG1W4 44452197 IC50 = 420 nM T79062 C5DNK1 44452199 IC50 = 710 nM T79062 CA3Y7E 44452217 IC50 = 48 nM T79062 CFUM27 44452219 IC50 = 1100 nM T79062 CAI2D5 44452221 IC50 = 690 nM T79062 CVAU93 44452222 IC50 = 460.26 nM T79062 CD0CQ5 44452223 IC50 = 1400 nM T79062 C6TN5J 44452224 IC50 = 79.98 nM T79062 CD8AJ3 44452243 IC50 = 79 nM T79062 C69RGK 44452244 IC50 > 10000 nM T79062 C1HEZ2 44452245 IC50 = 110 nM T79062 CJD35V 44452246 IC50 = 84.92 nM T79062 C23DZP 44452247 IC50 = 159.96 nM T79062 CLPR24 44452249 IC50 = 449.78 nM T79062 CJY18I 44452251 IC50 = 1099.01 nM T79062 C0G6ZC 44452273 IC50 = 28.97 nM T79062 CD5IY1 44452274 IC50 = 210 nM T79062 CX4DR9 44452275 IC50 = 590 nM T79062 CDLB90 44452276 IC50 = 1500 nM T79062 C6CT8L 44452277 IC50 = 109.9 nM T79062 CF5G0O 44452278 IC50 = 130 nM T79062 CKU52M 44452279 IC50 = 639.73 nM T79062 CP4M7B 44452298 IC50 = 590.2 nM T79062 CMBT16 44452301 IC50 = 939.72 nM T79062 CFH72P 44452302 IC50 = 2398.83 nM T79062 CRE1X3 44452305 IC50 = 95 nM T79062 C4B8JL 44452324 IC50 = 74 nM T79062 C0B3LC 44452327 IC50 = 75 nM T79062 C6SF7C 44452328 IC50 = 449.78 nM T79062 C6V1WM 44452329 IC50 = 400 nM T79062 CQX6I3 44452331 IC50 = 650 nM T79062 C8HI7Q 44452332 IC50 = 730 nM T79062 CCHJ25 44452357 IC50 = 349.95 nM T79062 C5U3VQ 44452359 IC50 = 920 nM T79062 C2QBM9 44452362 IC50 = 7294.58 nM T79062 CZL97F 44455426 Ki = 116 nM T79062 CYS7T4 44455943 Ki = 73 nM T79062 C6BFI0 44456033 Ki = 6 nM T79062 CG91RD 44456395 Ki = 12.4 nM T79062 C12XGE 44456400 Ki = 1148.15 nM T79062 C13YGE 44460471 Ki = 31 nM T79062 CHA10N 44460639 Ki = 166 nM T79062 C7KP0I 44460641 Ki = 125 nM T79062 C7HNZ8 44460642 Ki = 140 nM T79062 CVF5C3 44460669 Ki = 109 nM T79062 CQ2ID1 44460701 Ki = 139 nM T79062 C9DUW7 44460708 Ki = 10 nM T79062 C4YB7R 44460724 Ki = 109 nM T79062 CN6K9F 44460725 Ki = 23 nM T79062 CF6A9J 44460738 Ki = 34 nM T79062 C46ZGA 44460739 Ki = 158 nM T79062 CV0PU6 44460744 Ki = 182 nM T79062 C8P1MO 44460759 Ki = 288 nM T79062 CCL32X 44460808 Ki = 88 nM T79062 C9UW7I 44460917 Ki = 70 nM T79062 C3PK8D 44460918 Ki = 145 nM T79062 CSI97R 44460980 Ki = 70 nM T79062 CCX4G5 44461045 Ki = 17 nM T79062 C0RE6D 44461048 Ki = 9 nM T79062 CR6J9L 44461052 Ki = 163 nM T79062 C05GVU 44461064 Ki = 1573 nM T79062 C7G4MW 44461065 Ki = 10 nM T79062 CKE9C5 44461066 Ki = 16 nM T79062 C62CSN 44461069 Ki = 37 nM T79062 CK5SR9 44461070 Ki = 14 nM T79062 C4DL5C 44469677 IC50 > 10000 nM T79062 CEX18U 44517732 Ki = 195 nM T79062 C3I9NZ 44517733 Ki = 339 nM T79062 C3D4HR 44537940 Ki > 5000 nM T79062 CJ7U3K 44554227 Ki > 5000 nM T79062 CM0I1P 44554393 Ki > 5000 nM T79062 CNHA47 44554395 Ki > 5000 nM T79062 C0NGQ3 44575261 IC50 > 150000 nM T79062 CEGL62 44576914 IC50 > 10000 nM T79062 CW8OI7 44576978 IC50 = 103 nM T79062 C1S9PB 44576979 IC50 > 10000 nM T79062 C0TN9C 44576980 IC50 > 10000 nM T79062 C3R0YE 44577013 IC50 > 10000 nM T79062 CRCH48 44582675 Ki = 59 nM T79062 CEJ4R8 44582676 Ki = 210 nM T79062 CZGP86 44582677 Ki = 5170 nM T79062 C5QB4K 44582678 Ki = 498 nM T79062 C01RCI 44582705 Ki = 731 nM T79062 CXL25V 44582706 Ki > 10000 nM T79062 C8MR1X 44582707 Ki = 6241 nM T79062 C4IT1N 44582708 Ki = 2862 nM T79062 CB0S4Z 44592109 IC50 > 1000 nM T79062 C6KTM4 45028192 Ki = 9549.93 nM T79062 C0DLU3 45109862 IC50 = 456 nM T79062 CGB2Z0 45113400 Ki = 42 nM T79062 CV1F6P 45268647 Ki = 276 nM T79062 CGZ08S 45269494 Ki = 198 nM T79062 CR2QP3 45272864 Ki = 177 nM T79062 CX15SL 45272891 Ki = 140 nM T79062 CTD71C 45273807 Ki = 161 nM T79062 C13MCR 45273816 Ki = 150 nM T79062 CZ71RN 45278805 IC50 = 333 nM T79062 CZN6M7 45278882 IC50 = 408 nM T79062 C6NT3Q 45278883 IC50 = 493 nM T79062 CS5BA4 45278886 IC50 = 524 nM T79062 C0CHF4 45482789 IC50 > 10000 nM T79062 CH90CZ 45488126 Ki > 500 nM T79062 CG9U2R 45488130 Ki > 500 nM T79062 C7N4GP 45488138 Ki > 500 nM T79062 CH29KP 45488139 Ki > 500 nM T79062 CDAJ27 45488143 Ki > 500 nM T79062 CZYC01 45488151 Ki > 500 nM T79062 C8PH0Y 45488152 Ki > 500 nM T79062 CC2OU0 45488156 Ki > 500 nM T79062 CL4G8T 45488165 Ki > 500 nM T79062 C5NDO6 45488166 Ki > 500 nM T79062 C0GMN4 45488171 Ki > 500 nM T79062 C3ZAL4 45488172 Ki > 500 nM T79062 C3PYL9 45488174 Ki > 500 nM T79062 CFT7C5 45488175 Ki > 500 nM T79062 CX1A2N 45488179 Ki > 500 nM T79062 CA8I7U 45488180 Ki > 500 nM T79062 C01QBM 45488181 Ki > 500 nM T79062 COX47A 45488183 Ki > 500 nM T79062 C8ETO2 45488184 Ki > 500 nM T79062 C5FQ4S 46224879 Ki = 0.2089 nM T79062 CXUL12 46232559 IC50 = 195 nM T79062 CU2RG8 46232560 IC50 = 456 nM T79062 C9RQ8U 46232586 IC50 = 110 nM T79062 C2B3ZP 46232587 IC50 = 87 nM T79062 C3I8TO 46232588 IC50 = 567 nM T79062 COW9V6 46232589 IC50 = 172 nM T79062 CGV2J5 46232620 IC50 = 678 nM T79062 CWHG97 46232621 IC50 = 980 nM T79062 CUQW08 46232622 IC50 = 1236 nM T79062 C5REP7 46232623 IC50 = 500 nM T79062 C2QOW0 46232652 IC50 = 888 nM T79062 C9I7XS 46232653 IC50 = 1508 nM T79062 C5D0BH 46232654 IC50 = 419 nM T79062 C5PAL9 46232689 IC50 = 24 nM T79062 CT5C0M 46232690 IC50 = 160 nM T79062 CF53BL 46232691 IC50 = 442 nM T79062 CE1ID7 46232729 IC50 = 2296 nM T79062 CN0CO9 46232730 IC50 = 152 nM T79062 C0VXA5 46232731 IC50 = 334 nM T79062 C1C4OF 46232732 IC50 = 147 nM T79062 CMR8O9 46232770 IC50 = 500 nM T79062 CTY9H7 46232771 IC50 = 121 nM T79062 C5TBE8 46232772 IC50 = 316 nM T79062 COH03R 46232773 IC50 = 124 nM T79062 CZ2W7X 46232817 IC50 = 93 nM T79062 C0N4YP 46232818 IC50 = 117 nM T79062 CTJ89I 46232819 IC50 = 188 nM T79062 CS98DM 46232820 IC50 = 342 nM T79062 C8P3HD 46232858 IC50 = 49.6 nM T79062 CP04TS 46232859 IC50 = 749 nM T79062 C8W0IJ 46232860 IC50 = 12.3 nM T79062 CF5M2T 46232861 IC50 = 6.3 nM T79062 C21CHG 46232975 IC50 = 35.3 nM T79062 CO41KX 46232976 IC50 = 657 nM T79062 CIK94R 46232977 IC50 = 316 nM T79062 CB67ST 46232978 IC50 = 363 nM T79062 CRU0F7 46233014 IC50 = 526 nM T79062 C7W5TE 46233349 Ki = 2240 nM T79062 C10LFM 46233350 Ki = 128 nM T79062 C5NT9Y 46233351 Ki = 1614 nM T79062 C4T3HL 46233352 Ki = 26 nM T79062 C75PCA 46233382 Ki = 669 nM T79062 CV2FO0 46233383 Ki = 1429 nM T79062 C0QBP6 46233384 Ki > 10000 nM T79062 CL54OR 46233385 Ki > 10000 nM T79062 C3RH1V 46233448 Ki > 10000 nM T79062 C8USF7 46233449 Ki = 1485 nM T79062 C69MQR 46233450 Ki = 0.3 nM T79062 CNGP15 46233483 Ki > 10000 nM T79062 C42SVX 46700866 IC50 > 10000 nM T79062 CD0K6E 46700867 IC50 = 5600 nM T79062 C5TC2S 46830335 IC50 > 10000 nM T79062 C1K7FL 46830336 IC50 > 10000 nM T79062 C1N4KX 46842383 IC50 > 10000 nM T79062 CC62SX 46866711 IC50 = 2874 nM T79062 C03LTM 46869265 Ki = 220000 nM T79062 CB8GE1 46884818 IC50 > 10000 nM T79062 C4MQ0A 46884856 IC50 > 10000 nM T79062 CCNT25 46884898 IC50 > 10000 nM T79062 C3MSG2 46885027 IC50 > 10000 nM T79062 CB7XI0 46885213 IC50 > 10000 nM T79062 CY28OS 47556338 Ki = 888 nM T79062 C2LZJ0 49783209 Ki = 5702 nM T79062 C57SMG 49783415 Ki > 10000 nM T79062 C0TG6I 49783419 Ki > 10000 nM T79062 CR40BA 49836386 IC50 > 1000 nM T79062 C4R2YS 49850567 Ki = 199.53 nM T79062 C07JTU 49850570 Ki = 39.81 nM T79062 CK68QR 49850672 Ki = 25.12 nM T79062 CN5XR1 49850772 Ki = 125.89 nM T79062 CR4EZ0 49850870 Ki = 100 nM T79062 C5K4EC 49850872 Ki = 63.1 nM T79062 C8AW0R 49850874 Ki = 79.43 nM T79062 C6OQV2 49862237 Ki = 15 nM T79062 C9KIU1 49864289 IC50 = 3038 nM T79062 CHO9C0 49864292 IC50 = 2044 nM T79062 C90MTG 49864602 IC50 = 1006 nM T79062 C5BCS4 49864722 IC50 = 4425 nM T79062 CKZO79 49864723 IC50 = 3865 nM T79062 C74LZS 49864724 IC50 = 2059 nM T79062 C2RY0J 50878551 Ki = 16.98 nM T79062 C1W6TV 50898777 Ki > 10000 nM T79062 CXMZ73 50898778 Ki > 10000 nM T79062 CX48AD 51002362 Ki = 1956 nM T79062 C8TA1J 51003550 IC50 > 10000 nM T79062 CQ1UJ7 51003551 IC50 = 2007 nM T79062 CGMI37 51003586 IC50 > 10000 nM T79062 CE4KP1 51050257 Ki > 10000 nM T79062 CT3HG0 52952098 Ki > 100000 nM T79062 CDM75V 52952099 Ki = 14125.38 nM T79062 CR0ES9 52952100 Ki > 100000 nM T79062 CI9BF4 52952200 Ki = 91201.08 nM T79062 C31KMJ 52952201 Ki > 100000 nM T79062 CG4AW2 52952202 Ki = 15135.61 nM T79062 C3KZA4 52952203 Ki > 100000 nM T79062 C0MC9X 52952204 Ki > 100000 nM T79062 CT7A6Q 52952304 Ki > 100000 nM T79062 CR96JZ 52952305 Ki > 100000 nM T79062 CN70EP 52952306 Ki > 100000 nM T79062 CUI85Q 52952307 Ki = 9120.11 nM T79062 CJ94KO 52952308 Ki = 7244.36 nM T79062 C39XRU 52952309 Ki = 4786.3 nM T79062 C53DTC 52952419 Ki = 53703.18 nM T79062 COZ2U3 52952420 Ki = 12589.25 nM T79062 CG0L5I 52952421 Ki = 8709.64 nM T79062 CHC1S3 52952422 Ki = 263.03 nM T79062 CP37CU 52952423 Ki > 100000 nM T79062 C6LRO4 52952424 Ki = 27542.29 nM T79062 CMJ62D 53245590 Ki = 930 nM T79062 CGY45S 53248361 Ki = 161 nM T79062 CE9L8G 53248365 Ki = 50 nM T79062 C61DNP 53320009 IC50 = 143 nM T79062 C9ZDR5 53320010 IC50 = 620 nM T79062 CQLK01 53322638 IC50 > 10000 nM T79062 C32YWL 53324045 Ki = 326 nM T79062 CY28UP 53324535 Ki = 14 nM T79062 CRQF15 53325242 Ki = 969 nM T79062 C70WHV 53361627 Ki = 404 nM T79062 CU4B6N 53370045 Ki = 125 nM T79062 CKQ6A3 53376040 Ki = 739 nM T79062 C65CWD 53377240 Ki > 10000 nM T79062 CSGU70 53377324 Ki = 418 nM T79062 CG24AT 53381002 Ki = 1985 nM T79062 CMOZ61 53475319 Ki = 770 nM T79062 C0J8XZ 54598062 Ki = 26 nM T79062 C8SJ1Z 54758201 Ki = 107 nM T79062 C6G2AC 54758202 Ki = 72 nM T79062 CU6HI4 54758203 Ki = 96 nM T79062 C5KGQ3 54758204 Ki = 11 nM T79062 CS6PX1 54758293 Ki = 5.1 nM T79062 C6X3OI 54758294 Ki = 139 nM T79062 CS9L0P 54758295 Ki = 4 nM T79062 CUD7N0 54758296 Ki = 52 nM T79062 C1H2GP 54758297 Ki = 16 nM T79062 CG3UJ4 54758298 Ki = 6.7 nM T79062 C89NYL 54758391 Ki = 40 nM T79062 CTH56O 54758392 Ki = 13 nM T79062 CAZ5T6 54764323 Ki = 13 nM T79062 COZ82F 55479093 Ki = 155 nM T79062 CW89BT 56595402 Ki > 1000 nM T79062 C4C3XQ 56595529 Ki > 1000 nM T79062 C6W1RA 56649648 Ki = 132 nM T79062 C2SW7J 56649649 Ki = 77 nM T79062 CQTR49 56649650 Ki = 97 nM T79062 CH37LU 56663451 IC50 > 10000 nM T79062 CJKO58 56852956 Ki = 338.84 nM T79062 C1ZG7A 56933434 Ki = 0.6 nM T79062 CO0N2W 56943599 Ki = 6.7 nM T79062 C3DF5Z 56943600 Ki = 3.2 nM T79062 C19BDH 56943695 Ki = 10 nM T79062 CS7K3T 56943891 Ki = 6.9 nM T79062 CZ4L3S 56944082 Ki = 0.1 nM T79062 C5NI3K 56944086 Ki = 67 nM T79062 C37BYO 56944186 Ki = 5.1 nM T79062 C9UOZ6 56944189 Ki = 5.9 nM T79062 CH7V9J 56944190 Ki = 5.1 nM T79062 CE49MC 56944191 Ki = 4.4 nM T79062 CX2RP5 56944287 Ki = 15 nM T79062 CB0P9N 56944383 Ki = 1.6 nM T79062 CEQ7I3 56944384 Ki = 1.3 nM T79062 CHWI01 56944473 Ki = 13 nM T79062 C6Y4ZQ 56944564 Ki = 1.8 nM T79062 C3B0MZ 56944565 Ki = 1.6 nM T79062 CI4KW0 56944664 Ki = 1.1 nM T79062 C39YHD 56944665 Ki = 0.8 nM T79062 C1W3GL 56944666 Ki = 1.4 nM T79062 C7J4UT 56944667 Ki = 1.5 nM T79062 CZT80U 56944668 Ki = 0.8 nM T79062 CTW2F5 56944763 Ki = 0.4 nM T79062 C50WEX 56944764 Ki = 1.1 nM T79062 CX0ZW2 56944859 Ki = 1.3 nM T79062 C1ST9U 56944860 Ki = 140 nM T79062 CQKL90 56944861 Ki = 110 nM T79062 CS5J6Y 56944862 Ki = 90 nM T79062 CFLB40 56944863 Ki = 65 nM T79062 C53OTR 56944864 Ki = 70 nM T79062 C5T3RI 56944951 Ki = 18 nM T79062 CR6H7U 56944952 Ki = 10 nM T79062 C1Y2RP 56944953 Ki = 6 nM T79062 C1BH7I 56944954 Ki = 2 nM T79062 CTK9I8 56944955 Ki = 29 nM T79062 CCF1A5 56944956 Ki = 2 nM T79062 C2YVT8 56945042 Ki = 51 nM T79062 CNI2G3 56945043 Ki = 17 nM T79062 CF9V3Q 56945045 Ki = 33 nM T79062 CE4S5M 56945046 Ki = 38 nM T79062 C1TC7Q 56963799 Ki > 10000 nM T79062 C3ZG6J 57325520 Ki = 56 nM T79062 CDK7B0 57325521 Ki = 47 nM T79062 CR9MZ4 57384073 Ki = 16 nM T79062 CO7BG0 57390335 Ki = 335 nM T79062 CP05DB 57390336 Ki = 235 nM T79062 C1TH4R 57390337 Ki = 41 nM T79062 CATM39 57390694 Ki = 2060 nM T79062 C6S0IE 57390695 Ki = 2810 nM T79062 C83GWU 57391158 Ki = 604 nM T79062 CPE8N4 57391622 Ki = 68 nM T79062 CHG51U 57391624 Ki = 36 nM T79062 CIHJ73 57392107 Ki = 55 nM T79062 CY02VL 57392108 Ki = 38 nM T79062 C93QRW 57393876 Ki = 267 nM T79062 CUF40C 57393877 Ki = 334 nM T79062 CR7FB5 57393878 Ki = 1255 nM T79062 C7VFQ3 57394663 Ki = 50 nM T79062 CEW0O4 57395084 Ki = 88 nM T79062 CL96RC 57395086 Ki = 25 nM T79062 CSI7X2 57395597 Ki = 360 nM T79062 CJ15YT 57395598 Ki = 228 nM T79062 CK53EW 57395599 Ki = 37 nM T79062 C51GCK 57396417 Ki = 207 nM T79062 CZ2SJ8 57396419 Ki = 40 nM T79062 CZ8KA2 57396855 Ki = 381 nM T79062 CN7QE4 57396857 Ki = 334 nM T79062 C2Q6CJ 57397410 Ki = 132 nM T79062 CFQA13 57397411 Ki = 995 nM T79062 C7W5XA 57398619 Ki = 113 nM T79062 CFT56H 57399088 Ki = 3010 nM T79062 CGX5Q1 57399089 Ki = 79 nM T79062 CTF76G 57399090 Ki = 156 nM T79062 C0XFB2 57399091 Ki = 90 nM T79062 CI6ET3 57399092 Ki = 29 nM T79062 CMX4K5 57399093 Ki = 33 nM T79062 CJ41PW 57399432 Ki = 413 nM T79062 CAN0W7 57399866 Ki = 145 nM T79062 C9BG7C 57399868 Ki = 126 nM T79062 C5HGO2 57400281 Ki = 69 nM T79062 CT7Q3E 57400828 Ki = 506829 nM T79062 CFBP89 57400829 Ki = 1420 nM T79062 C3D1UP 57400830 Ki = 187 nM T79062 C5GPJ0 57401515 Ki = 210 nM T79062 CG8MF3 57401516 Ki = 353 nM T79062 CZX05B 57401706 Ki = 291 nM T79062 CN9J5I 57402588 Ki = 224 nM T79062 C92HON 57402951 Ki = 356 nM T79062 CX0B5M 57403525 Ki = 1042 nM T79062 C3A1YW 57403839 Ki = 310 nM T79062 CA10YX 57403841 Ki = 335 nM T79062 CYSV60 60165411 Ki = 337 nM T79062 CB9GC6 60165412 Ki = 62.6 nM T79062 CI5PM3 60165413 Ki = 107 nM T79062 C2Q5VD 60165416 Ki = 329 nM T79062 C9JL3F 60165418 Ki = 228.9 nM T79062 C31PEN 60165535 Ki = 35.6 nM T79062 CP60YF 60165537 Ki = 211 nM T79062 C85OTH 60165541 Ki = 425.8 nM T79062 CJO91V 60165543 Ki = 2467 nM T79062 CJDC53 60165545 Ki = 242 nM T79062 C3K5JN 60165681 Ki = 2917 nM T79062 C5RUP6 60167166 Ki = 790 nM T79062 CRH49P 60167309 Ki = 983 nM T79062 COHK72 60167451 Ki = 125.89 nM T79062 C30SVG 60167452 Ki = 512.86 nM T79062 CB4HT7 60195992 Ki = 109 nM T79062 C4Q6LO 60195993 Ki = 1.9 nM T79062 C04CRJ 60195994 Ki = 93 nM T79062 C4BG3H 60195995 Ki > 5000 nM T79062 C87FDE 60195996 Ki = 7 nM T79062 C6VWY1 60196073 Ki = 13 nM T79062 CM92UX 60196074 Ki = 23 nM T79062 C18AVJ 60196075 Ki = 80 nM T79062 CZN64D 60196076 Ki = 96 nM T79062 CIN29U 60196077 Ki = 7.1 nM T79062 C3LTC1 60196078 Ki = 8.2 nM T79062 C7WLN1 60196079 Ki = 6.9 nM T79062 C5N3SG 60196080 Ki = 1.4 nM T79062 C6AUO2 66800823 Ki = 25 nM T79062 C34ACQ 66800909 Ki = 2 nM T79062 CGT9E6 66800910 Ki = 6.3 nM T79062 C0QY7D 66800916 Ki = 4.6 nM T79062 CM58FG 66800926 Ki = 200 nM T79062 CQ43WD 66800934 Ki = 19 nM T79062 CK0I5J 66800939 Ki = 1.5 nM T79062 C0X2SF 66800942 Ki = 3.8 nM T79062 CN30YT 66800947 Ki = 9 nM T79062 CZ3MR6 66800959 Ki = 180 nM T79062 C92CMO 66800965 Ki = 91 nM T79062 CFPK92 66800991 Ki = 6.3 nM T79062 C13GMO 66801000 Ki = 13 nM T79062 CZ1TF9 66801018 Ki = 2.6 nM T79062 CBO9U3 66801028 Ki = 8.8 nM T79062 C3K8DC 66801052 Ki = 80 nM T79062 CA4DM3 66801062 Ki = 4.1 nM T79062 C2OUX9 66801107 Ki = 1.7 nM T79062 C4J5RZ 66801115 Ki = 54 nM T79062 C1H8BS 66801116 Ki = 41 nM T79062 C4JGC6 66801120 Ki = 18 nM T79062 CX2GN1 66801139 Ki = 0.9 nM T79062 C1NG8S 66801140 Ki = 5.3 nM T79062 CR7OW6 66801158 Ki = 0.8 nM T79062 CJU53X 66801160 Ki = 9.5 nM T79062 CH3BJ8 66801167 Ki = 0.5 nM T79062 C0AV5M 66801173 Ki = 9.9 nM T79062 C0V9EF 66801186 Ki = 3.2 nM T79062 CTHY41 66801210 Ki = 0.7 nM T79062 CSD67P 66801225 Ki = 4.3 nM T79062 C8J3YU 66801226 Ki = 9.9 nM T79062 CX45OZ 66801229 Ki = 1.5 nM T79062 C1S0EV 66801230 Ki = 3.2 nM T79062 C7S1KY 66801234 Ki = 0.9 nM T79062 CB53AV 66801246 Ki = 14 nM T79062 C3F1TZ 66801251 Ki = 34 nM T79062 CF8O9U 66801259 Ki = 57 nM T79062 C2Q9FS 66801263 Ki = 0.7 nM T79062 C7Y9VP 66801267 Ki = 2500 nM T79062 CED17M 66801271 Ki = 0.9 nM T79062 C41VYW 66801295 Ki = 14 nM T79062 C2FYL1 66801333 Ki = 180 nM T79062 CS75LK 66801335 Ki = 29 nM T79062 CR2N0J 66801344 Ki = 15 nM T79062 CDH7S9 66801346 Ki = 1.2 nM T79062 CGC4U6 66801354 Ki = 120 nM T79062 CY4FM5 66801379 Ki = 3.4 nM T79062 C3RX4C 66801425 Ki = 120 nM T79062 C7JD0I 66801429 Ki = 24 nM T79062 CN8OU1 66801430 Ki = 150 nM T79062 C93EGP 66801455 Ki = 4.1 nM T79062 COR1H8 66801528 Ki = 80 nM T79062 C1F3YV 66801537 Ki = 69 nM T79062 CIRW86 66801551 Ki = 0.2 nM T79062 C75WXP 66801561 Ki = 240 nM T79062 C8H5PD 66801565 Ki = 1.3 nM T79062 CT5SP8 66801605 Ki = 9 nM T79062 C8MH0I 66801613 Ki = 20 nM T79062 CC8JV6 66801624 Ki = 520 nM T79062 C3EI2F 66801625 Ki = 150 nM T79062 C49XBJ 66801673 Ki = 34 nM T79062 C0XG6B 66801701 Ki = 380 nM T79062 C42EBQ 66801837 Ki = 610 nM T79062 CW3AI2 66803474 Ki = 0.6 nM T79062 CPKH06 66803497 Ki = 12 nM T79062 CNJE57 66803500 Ki = 61 nM T79062 CN6FZ1 66803595 Ki = 1 nM T79062 C1LEH8 67268994 Ki = 30 nM T79062 CLA7F3 68281136 Ki = 23 nM T79062 C84MZH 68281137 Ki = 270 nM T79062 CR5KY1 71061607 Ki = 18 nM T79062 C72XPZ 71061659 Ki = 23.8 nM T79062 CKE2Y4 71061750 Ki = 26.1 nM T79062 CD1ET2 71061756 Ki = 23.5 nM T79062 C5KM2W 71061887 Ki = 11.2 nM T79062 C0D5SC 71062035 Ki = 15.2 nM T79062 CNQ65S 71062123 Ki = 12.7 nM T79062 CC43QK 71151588 Ki = 180 nM T79062 C3PUX5 71449549 Ki = 27 nM T79062 CN82LY 71449550 Ki = 311 nM T79062 C40DOC 71449627 Ki = 276 nM T79062 C8U6NR 71449628 Ki = 709 nM T79062 C7Y6LC 71449629 Ki = 7 nM T79062 C91SZN 71449641 Ki = 13 nM T79062 C2GCN7 71449642 Ki = 121 nM T79062 CQN93U 71449643 Ki = 7 nM T79062 CEJ3B4 71449644 Ki = 16 nM T79062 C5SAJ1 71449645 Ki = 28 nM T79062 C3XNC2 71450247 Ki = 1914 nM T79062 C9VZ8J 71450550 Ki = 3505 nM T79062 C2IXB6 71451344 Ki = 409 nM T79062 C7DCR4 71451345 Ki = 1672 nM T79062 CC6QP7 71451441 Ki = 161 nM T79062 CHT21G 71451454 Ki = 2222 nM T79062 C2QZL4 71451455 Ki = 78 nM T79062 CXI5Q2 71451456 Ki = 2375 nM T79062 CKJZ57 71451457 Ki = 29 nM T79062 C0F1HU 71451458 Ki = 15 nM T79062 CTZ24N 71451459 Ki = 6 nM T79062 C70JUP 71451460 Ki = 4 nM T79062 C4NDR3 71452382 Ki = 6259 nM T79062 C6ZWV2 71452383 Ki = 6873 nM T79062 CGO4M1 71453156 Ki = 815 nM T79062 C6EFP9 71453157 Ki = 391 nM T79062 CUK2P5 71453252 Ki = 12 nM T79062 CKI58Z 71453278 Ki = 21 nM T79062 C1QM8D 71453279 Ki = 58 nM T79062 C6O4KT 71453280 Ki = 9 nM T79062 CL49VI 71453281 Ki = 4 nM T79062 CGXT64 71453282 Ki = 12 nM T79062 CQ3XC8 71454898 Ki = 865 nM T79062 CWY38Z 71454899 Ki = 1188 nM T79062 CGO13Q 71454997 Ki = 20 nM T79062 C0K1JV 71454998 Ki = 46 nM T79062 C3JF1D 71454999 Ki = 0.3 nM T79062 C2QZ1N 71455000 Ki = 7 nM T79062 C6FE5D 71455001 Ki = 293 nM T79062 C4L0JN 71455002 Ki = 2 nM T79062 C8YH0J 71455083 Ki = 60 nM T79062 CAQF34 71455625 Ki = 1945 nM T79062 C6G2HC 71455894 Ki = 3647 nM T79062 C5O6LT 71456677 Ki = 1500 nM T79062 CLX0G4 71456770 Ki = 85 nM T79062 CE19SD 71456779 Ki = 97 nM T79062 CWR40I 71456780 Ki = 2195 nM T79062 CZUX67 71456781 Ki = 10 nM T79062 CZ17FC 71456782 Ki = 9 nM T79062 CKF09U 71456783 Ki = 16 nM T79062 CJKV72 71456784 Ki = 10 nM T79062 C7MNB5 71457264 Ki = 6371 nM T79062 CMJ1O9 71457409 Ki = 1018 nM T79062 CVI7S2 71457690 Ki = 2447 nM T79062 CG83QI 71458516 Ki = 334 nM T79062 CE6OC0 71458622 Ki = 1144 nM T79062 CZ8L0D 71458623 Ki = 17 nM T79062 CW79AY 71458624 Ki = 59 nM T79062 C2XV5L 71458625 Ki = 5 nM T79062 CUAC42 71458626 Ki = 5 nM T79062 C37EBC 71458647 Ki = 60 nM T79062 CM6OP1 71458648 Ki = 1362 nM T79062 CRGE05 71458649 Ki = 1438 nM T79062 CJN4S1 71458650 Ki = 14 nM T79062 CNT5J9 71458651 Ki = 10 nM T79062 C3NAM7 71458652 Ki = 11 nM T79062 CS83IF 71459269 Ki = 150 nM T79062 CK5T4P 71459604 Ki = 3601 nM T79062 CG0WO9 71459954 Ki = 329 nM T79062 CMW0T6 71460453 Ki = 93 nM T79062 C9W7CF 71460454 Ki = 3372 nM T79062 C09VSE 71460455 Ki = 1104 nM T79062 CBU8J7 71460456 Ki = 2224 nM T79062 CT17XB 71460468 Ki = 178 nM T79062 C63YLA 71461049 Ki = 3473 nM T79062 CJD96I 71461050 Ki = 384 nM T79062 CZ6G8V 71462064 Ki = 2674 nM T79062 CI0K3L 71462065 Ki = 415 nM T79062 CD0G8Q 71462066 Ki = 407 nM T79062 CK5JC7 71462067 Ki = 329 nM T79062 C42IZX 71462068 Ki = 873 nM T79062 CB30LT 71462154 Ki = 204 nM T79062 C7Y1XU 71462155 Ki = 427 nM T79062 CLS2A6 71462156 Ki = 1108 nM T79062 C7AX1Q 71462178 Ki = 41 nM T79062 C1CS0Z 71462179 Ki = 27 nM T79062 C4P3JU 71462776 Ki = 153 nM T79062 C3GUQ2 71462777 Ki > 10000 nM T79062 CT2ME3 71574204 Ki = 21 nM T79062 C3SXR5 71574206 Ki = 46 nM T79062 C2YRI9 71574208 Ki = 31 nM T79062 C62RWV 71574210 Ki = 12 nM T79062 CKC53S 71574212 Ki = 30 nM T79062 CNV42M 71574298 Ki = 41 nM T79062 C9PGQ1 71574300 Ki = 124 nM T79062 C2LXH5 71574302 Ki = 31 nM T79062 C2YPB8 71574304 Ki = 27 nM T79062 CK7GM0 71574306 Ki = 56 nM T79062 C7EQ2F 71602523 Ki = 537 nM T79062 C29INM 71602524 Ki > 10000 nM T79062 CK2C5Q 71602525 Ki > 10000 nM T79062 C1T0VP 71602526 Ki > 10000 nM T79062 C4BFZ0 71602581 Ki > 10000 nM T79062 C82MIC 71602582 Ki > 10000 nM T79062 C69MFB 71602583 Ki = 432 nM T79062 CG21CD 71602584 Ki > 10000 nM T79062 CQZ2O3 71602585 Ki > 10000 nM T79062 C9UE3T 71602586 Ki = 1850 nM T79062 C6B4VK 71602587 Ki = 1737.8 nM T79062 C9XWR8 71602639 Ki = 1200 nM T79062 CH91JF 71602640 Ki = 2754.23 nM T79062 C2KRC8 71602641 Ki > 10000 nM T79062 C1I9AS 71602642 Ki > 10000 nM T79062 CW3Z9S 71602643 Ki > 10000 nM T79062 C6MH1U 71602644 Ki > 10000 nM T79062 CKR10Z 71602687 Ki = 658 nM T79062 C3ZQ5D 71602688 Ki = 295.12 nM T79062 CJ89YE 71602689 Ki = 218.78 nM T79062 C6L3DJ 71602690 Ki = 199.53 nM T79062 C2ABS7 71602691 Ki = 309.03 nM T79062 CI86QM 71602692 Ki = 42.66 nM T79062 CC45VZ 71602739 Ki = 77 nM T79062 CXP3V8 71602740 Ki = 45.71 nM T79062 CVL36N 71678345 Ki = 1659.59 nM T79062 C0PF3I 71678857 Ki = 15 nM T79062 C0W2YA 71727193 Ki = 195 nM T79062 C79TLS 71727194 Ki = 16950 nM T79062 CFB10W 71727195 Ki = 13500 nM T79062 C6CIB5 71727196 Ki = 1145 nM T79062 C7Z3JS 71727308 Ki = 426 nM T79062 C3ATN5 72197484 IC50 = 1564 nM T79062 C20HSN 72197485 IC50 = 1059 nM T79062 CN8A5R 72197486 IC50 = 1003 nM T79062 CL3BF7 72197668 IC50 = 497 nM T79062 CUVJ59 72197845 Ki = 196 nM T79062 CIKU20 72198011 Ki = 345 nM T79062 COH95V 72198014 Ki = 589 nM T79062 C0WY2V 72198191 Ki = 1165 nM T79062 C7AOY4 72198754 IC50 = 62 nM T79062 C4M7KP 72198756 IC50 > 100 nM T79062 CWHF29 72547876 Ki = 43.7 nM T79062 CF47JC 72547878 Ki = 32.4 nM T79062 C12CIH 72548115 Ki = 26.1 nM T79062 C1UX8Q 72548117 Ki = 47.6 nM T79062 C4K1WO 72548349 Ki = 66.1 nM T79062 CWH6T3 72548703 IC50 = 0.39 nM T79062 C4T0SK 72549767 Ki = 186.5 nM T79062 CE4U6J 72549768 Ki = 64.5 nM T79062 C1QZ4F 72549986 Ki = 37.9 nM T79062 C17XNV 72549988 Ki = 43.7 nM T79062 CD7V6P 72550196 Ki = 36.5 nM T79062 C1SZ3K 72550200 Ki = 34.7 nM T79062 C62EFS 72550423 Ki = 34.7 nM T79062 CK0F1L 72550641 Ki = 46.6 nM T79062 C8Z0NM 72550642 Ki = 8.69 nM T79062 CL6W2Q 72550645 Ki = 15.9 nM T79062 CUH4Z3 72550864 Ki = 405.3 nM T79062 C9J4QU 72550865 Ki = 25.9 nM T79062 C8A3DU 72551082 Ki = 31.4 nM T79062 C78LYM 72698087 Ki > 10000 nM T79062 C63HPK 72698088 Ki > 10000 nM T79062 C7W4RH 72734860 Ki = 12.4 nM T79062 C8UCZ5 72734861 Ki > 100 nM T79062 CZ6SQ7 72734863 Ki = 42 nM T79062 C8JT6B 72734864 Ki = 144 nM T79062 CW4IB9 72734866 Ki > 1000 nM T79062 CY0AE3 72735038 Ki = 239 nM T79062 CAZ84Y 72735039 Ki > 1000 nM T79062 C0MT4E 72735040 Ki > 1000 nM T79062 C0CK8H 72735041 Ki > 100 nM T79062 CC6Q5R 72771081 Ki < 100 nM T79062 CC65OA 73213195 Ki = 199.53 nM T79062 CW83DK 73213196 Ki = 194.98 nM T79062 CCV91B 73346042 Ki = 17.2 nM T79062 CXM8O2 73347306 IC50 = 3100 nM T79062 C9X8GY 73347307 IC50 > 1000 nM T79062 C4ZM8R 73347582 Ki = 9.7 nM T79062 C6BS5L 73349361 Ki = 4423 nM T79062 CL38VQ 73351112 Ki > 1000 nM T79062 CC8I7X 73351903 IC50 = 1800 nM T79062 CG4M8P 73351905 IC50 = 3700 nM T79062 CAR7Z5 73354882 IC50 = 480 nM T79062 CET52A 73356443 IC50 = 690 nM T79062 CUB97Z 74538690 Ki = 35 nM T79062 C2E7QW 75201901 Ki = 7800 nM T79062 C8IDL3 75306277 Ki = 79.43 nM T79062 CX17RZ 76280896 Ki = 71 nM T79062 C45OSP 76284193 Ki = 53 nM T79062 C0CRJ1 76284452 Ki = 34.5 nM T79062 CS17IJ 76284453 Ki = 12.8 nM T79062 CH82JU 76284455 Ki = 45.2 nM T79062 CRO7Q9 76284721 Ki = 15.9 nM T79062 C4BIC2 76284724 Ki = 3.82 nM T79062 C0EKY7 76284725 Ki = 66.7 nM T79062 C3GXV8 76310809 Ki = 1200 nM T79062 C19EPD 76310810 Ki = 48 nM T79062 CK2X7A 76310812 Ki = 92 nM T79062 CXJG08 76314094 Ki > 1000 nM T79062 CN7GD5 76314435 Ki = 317 nM T79062 CLO9M1 76314437 Ki = 1920 nM T79062 CD8A5H 76318011 Ki = 6.9 nM T79062 C1Y9SX 76318012 Ki = 20 nM T79062 CEHK31 76321734 Ki = 4.5 nM T79062 C5F1XU 76321735 Ki = 4.5 nM T79062 CC8TR0 76321736 Ki = 70 nM T79062 C94VNF 76324975 Ki = 64.2 nM T79062 C18OSZ 76325346 Ki = 17 nM T79062 C62CZO 76325348 Ki = 27 nM T79062 COGC62 76325350 Ki = 18 nM T79062 C1Q5NC 76325352 Ki = 8.7 nM T79062 CZ6P1E 76328545 Ki > 1000 nM T79062 C0OI2M 76328889 Ki = 283 nM T79062 C51CME 76328891 Ki = 41 nM T79062 CBFE85 76328893 Ki = 62 nM T79062 C5WG9E 76328895 Ki = 60 nM T79062 C6OV4J 76328897 Ki = 65 nM T79062 CL83OY 76332574 Ki = 649 nM T79062 CN3QO1 76332576 Ki = 15 nM T79062 CDBS57 76332578 Ki = 34 nM T79062 C97OVP 76332580 Ki = 4440 nM T79062 C1LT6C 76332582 Ki = 3907 nM T79062 CP0D6T 76332584 Ki = 94 nM T79062 CW3AK0 76335863 Ki = 33.4 nM T79062 CYT34W 76336176 Ki = 33 nM T79062 C9XFL1 76336178 Ki = 18 nM T79062 C0GD2B 76336180 Ki = 20 nM T79062 CV90GC 76336182 Ki = 189 nM T79062 C51CXD 76336183 Ki = 54 nM T79062 CMG58X 76336185 Ki = 10.8 nM T79062 C28RIZ 76518514 Ki = 472 nM T79062 C9S0XK 86288947 Ki = 3 nM T79062 CEPC94 86288948 Ki = 3 nM T79062 CHE2U4 90178632 Ki = 16 nM T79062 CFDW68 90644074 Ki = 10 nM T79062 C0T8RE 90644075 Ki = 380 nM T79062 C2KE9G 90644076 Ki = 94 nM T79062 C1SOF5 90644077 Ki = 150 nM T79062 CIE9Z2 90644078 Ki = 900 nM T79062 C37CYS 90654670 Ki = 101 nM T79062 C0IQ5R 90654671 Ki = 51 nM T79062 CVG2C1 90654672 Ki = 78 nM T79062 CU0ON1 90654673 Ki = 111 nM T79062 CJR3Y9 90654674 Ki = 148 nM T79062 CO1H4U 90654675 Ki = 551 nM T79062 CAY64Z 90654676 Ki = 302 nM T79062 CH0R8B 90654677 Ki = 579 nM T79062 CRFB56 90654678 Ki = 476 nM T79062 CPR21O 90654679 Ki = 393 nM T79062 C6YLV3 90654680 Ki = 725 nM T79062 CGUY51 90654681 Ki = 223 nM T79062 CK8X4O 90654682 Ki = 295 nM T79062 CH8UQ9 90654683 Ki = 107 nM T79062 CTQ23Z 90654684 Ki = 95 nM T79062 C9Q2JW 90654685 Ki = 1196 nM T79062 C98TJR 90654686 Ki = 18 nM T79062 CG3OI7 90654687 Ki = 22 nM T79062 CKTV83 90654688 Ki = 28 nM T79062 CVK85U 90654689 Ki = 163 nM T79062 CLG75D 90654690 Ki = 153 nM T79062 C7T9HW 90654691 Ki = 495 nM T79062 C92BZL 90654692 Ki = 567 nM T79062 C6CD9R 90654693 Ki = 634 nM T79062 C6H9NV 90654694 Ki = 1199 nM T79062 CR74SD 90654695 Ki = 4151 nM T79062 C7VM4O 90654696 Ki = 1865 nM T79062 CGFU53 90654697 Ki = 1312 nM T79062 C7BEZ8 90654698 Ki = 3134 nM T79062 CZ3IM2 90654699 Ki = 478 nM T79062 C8TMK5 90654700 Ki = 1188 nM T79062 C7GK3C 90654701 Ki = 113 nM T79062 CN8BO1 90654702 Ki = 179 nM T79062 CHIW63 90654703 Ki = 108 nM T79062 C1SAW2 90654704 Ki = 50 nM T79062 CJG31T 90654831 Ki = 95 nM T79062 CMU45O 90654832 Ki = 77 nM T79062 C3C4BW 90654834 Ki = 157 nM T79062 C8QWR3 90654835 Ki = 34 nM T79062 C6ZR9L 90654837 Ki = 70 nM T79062 C0AC7R 90654839 Ki = 72 nM T79062 CKLG40 90654841 Ki = 122 nM T79062 C5JS8D 90654843 Ki = 135 nM T79062 C4VHZ6 90654845 Ki = 45 nM T79062 CG78PS 90654847 Ki = 172 nM T79062 CL39WP 90654849 Ki = 123 nM T79062 C0TVQ9 90654851 Ki = 46 nM T79062 C4I1CU 90654853 Ki = 31 nM T79062 CZ28YC 90654855 Ki = 78 nM T79062 CRO83N 90654857 Ki = 456 nM T79062 C72RKV 90656669 Ki = 20.8 nM T79062 CJ8H1R 90656670 Ki = 92.5 nM T79062 CSF25H 90656671 Ki = 90.1 nM T79062 CGD60Y 90656672 Ki = 12.1 nM T79062 C4H1SB 90656673 Ki = 81.4 nM T79062 CID83U 90656674 Ki = 161.4 nM T79062 C0VDH3 90656675 Ki = 252.1 nM T79062 CC1L7T 90656676 Ki = 57 nM T79062 CCQU80 90656678 Ki = 84.8 nM T79062 CNSW31 90656679 Ki = 161.2 nM T79062 CITS52 90656680 Ki = 179.2 nM T79062 C3GA5B 90656681 Ki = 111.7 nM T79062 C9SX5R 90656682 Ki = 10.1 nM T79062 CGEF35 90656683 Ki = 2.9 nM T79062 C76OIR 90656684 Ki = 434.2 nM T79062 CH9F4Q 90656685 Ki = 20 nM T79062 C8NB7D 90656686 Ki = 161.1 nM T79062 C13YLN 90656687 Ki = 39.6 nM T79062 CU82QN 90656688 Ki = 63.3 nM T79062 CNB76X 90656689 Ki = 77.9 nM T79062 CPQ46T 90656690 Ki = 108.8 nM T79062 C6QO1P 90656691 Ki = 13.2 nM T79062 C6TF2G 90656692 Ki = 8.1 nM T79062 CGP76X 90656694 Ki = 30 nM T79062 C3O2KS 90656695 Ki = 16.7 nM T79062 CYLZ26 90656696 Ki = 12 nM T79062 C9RH6O 90656697 Ki = 226 nM T79062 C5MP1J 90656699 Ki = 39.4 nM T79062 C5L9IQ 90656701 Ki = 95.6 nM T79062 C6NG4Q 90656703 Ki = 191 nM T79062 C63JKH 90656705 Ki = 137.5 nM T79062 C7NV3E 90656707 Ki = 242.1 nM T79062 CK6UO3 90656708 Ki = 310 nM T79062 C6N5CS 90656709 Ki = 40 nM T79062 CX49HI 90656710 Ki = 3.1 nM T79062 CRX47O 90656711 Ki = 11.6 nM T79062 CTHD25 90656712 Ki = 6.6 nM T79062 CID86Z 90656713 Ki = 12.8 nM T79062 C5Q8PH 90656714 Ki = 63.1 nM T79062 CS9E1R 90656715 Ki = 332 nM T79062 CCOV98 90664359 Ki = 10490 nM T79062 CA8B0H 90664441 Ki = 328 nM T79062 CP48OR 90664581 Ki = 612 nM T79062 C4MUI2 90664601 IC50 = 11 nM T79062 CXD5Q9 90664621 Ki = 17420 nM T79062 CP2MK1 90664692 Ki = 5800 nM T79062 CO9H3P 90664694 Ki = 153 nM T79062 CE6D5M 90664808 Ki = 296 nM T79062 CT7Z1V 90664944 Ki = 184 nM T79062 CHT7D5 90664962 IC50 = 6.8 nM T79062 CQCE48 90665063 Ki = 276 nM T79062 C4EQ5K 90665189 Ki = 484 nM T79062 C0J5YH 91864602 Ki = 3.548 nM T79062 CDWS84 91937906 Ki = 157 nM T79062 CEN10X 92042876 Ki = 5.2 nM T79062 CW6XB3 92042877 Ki = 15 nM T79062 CUQ6V0 92042918 Ki < 1000 nM T79062 CS62HU 101747513 Ki = 5.6 nM T79062 C4DG3V 102364516 Ki = 0.7 nM T79062 C4WDR8 109018769 Ki = 4.34 nM T79062 CD76TH 109026949 Ki = 52 nM T79062 C3DMI5 109026956 Ki = 29.5 nM T79062 C2G0WH 109026957 Ki = 23.5 nM T79062 CYB18Z 109027017 Ki = 26.2 nM T79062 C0M3CD 118051679 Ki = 42 nM T79062 CEMZ15 118464420 Ki = 401 nM T79062 CV2L6O 118464425 Ki = 516 nM T79062 CFNG86 118464427 Ki = 427 nM T79062 CMSN80 118626035 Ki = 19 nM T79062 CT3AI0 118626042 Ki = 75 nM T79062 CKNJ72 118626045 Ki = 23 nM T79062 CGB42Y 118626088 Ki = 66 nM T79062 C0XJT5 118626089 Ki = 19 nM T79062 CIE4C7 118626101 Ki = 4 nM T79062 C1NYS5 118626120 Ki = 142 nM T79062 CPG04R 118626121 Ki = 3 nM T79062 C3S5LJ 118626129 Ki = 1 nM T79062 CY3F0N 118626140 Ki = 97 nM T79062 CE07IQ 118626142 Ki = 4 nM T79062 C72OZY 118626161 Ki = 1 nM T79062 CY3E7S 118626169 Ki = 52 nM T79062 CHRB75 118626208 Ki = 349 nM T79062 CSN13R 118706278 Ki = 41 nM T79062 CIG56H 118706280 Ki > 1000 nM T79062 CF5ZR8 118706282 Ki = 14 nM T79062 CD1XJ5 118706284 Ki = 29 nM T79062 CL4Y6K 118706285 Ki = 4.1 nM T79062 C32KAS 118706287 Ki = 160 nM T79062 C1K5NC 118706290 Ki = 87 nM T79062 CGA0O1 118706292 Ki = 41 nM T79062 CA0V9U 118706294 Ki = 50 nM T79062 C0NSU5 118706296 Ki = 180 nM T79062 CFOE72 118706299 Ki = 57 nM T79062 C1DI6Y 118706301 Ki = 4.1 nM T79062 CH3Z8R 118706732 Ki = 4 nM T79062 CN4I3G 118706734 Ki = 2.3 nM T79062 C2Q4OP 118709739 Ki = 28 nM T79062 CZ68PL 118709740 Ki = 24 nM T79062 CSB25E 118709750 Ki = 917 nM T79062 CD4S9R 118709751 Ki = 882 nM T79062 CBP52O 118709752 Ki = 36 nM T79062 CO72SF 118709753 Ki = 29 nM T79062 CJQR81 118709754 Ki = 41 nM T79062 CPW1D5 118709755 Ki = 62 nM T79062 C1TMO7 118709756 Ki = 2.7 nM T79062 CZ9H5G 118711997 Ki = 22 nM T79062 CH9W0A 118713587 Ki = 36.48 nM T79062 CK43CN 118713588 Ki = 7.77 nM T79062 CL0TS7 118713589 Ki = 0.99 nM T79062 C4RD6F 118713590 Ki = 41.93 nM T79062 CIG13W 118713591 Ki = 46.83 nM T79062 CX5L1H 118713592 Ki = 1.72 nM T79062 CDWY84 118713593 Ki = 2.84 nM T79062 CO5S1I 118713594 Ki = 57.39 nM T79062 CI91US 118713595 Ki = 20 nM T79062 CW92LT 118713679 Ki = 5.9 nM T79062 C8P9YT 118713680 Ki = 5.16 nM T79062 CZ1K5R 118713681 Ki = 14.1 nM T79062 CH7ZE8 118713682 Ki = 2.96 nM T79062 CKX78H 118713683 Ki = 11.68 nM T79062 C5LSA7 118713684 Ki = 2.9 nM T79062 CPAI54 118713685 Ki = 45.57 nM T79062 C6U2LR 118713686 Ki = 7.58 nM T79062 CYA6E4 118713687 Ki = 7.73 nM T79062 CZ9UL2 118713688 Ki = 8.49 nM T79062 CI5XK3 118717210 Ki = 1.2 nM T79062 CYJQ09 118717212 Ki > 100 nM T79062 C1TSR8 118717214 Ki = 1.4 nM T79062 C7YX3Q 118717215 Ki = 0.6 nM T79062 CEZ4M6 118717216 Ki = 0.76 nM T79062 C1E4GL 118717218 Ki = 4.9 nM T79062 CSJ6N3 118717219 Ki = 1.8 nM T79062 C5LFW4 118717221 Ki = 1.7 nM T79062 CZ65GI 118717222 Ki = 1.3 nM T79062 C1F9ZM 118724639 Ki = 346 nM T79062 CGA86P 118728506 Ki = 168 nM T79062 C9PGE7 118728507 Ki = 357 nM T79062 CR4GE1 118728510 Ki = 30.1 nM T79062 C14LZH 118728511 Ki = 147 nM T79062 C14RAC 118728513 Ki = 68.4 nM T79062 CQK04P 118728514 Ki = 1464 nM T79062 CK9CG4 118728521 Ki = 307 nM T79062 C1N9JU 118728522 Ki = 1082 nM T79062 C1UZ8G 118728523 Ki = 35.8 nM T79062 CPCE84 118728524 Ki = 12.9 nM T79062 CBN06J 118728525 Ki = 6.88 nM T79062 CF3QE0 118728526 Ki = 143 nM T79062 CJG4Q1 118728527 Ki = 1650 nM T79062 C4NFW1 118728528 Ki = 88.5 nM T79062 CO8LF9 118728529 Ki = 213 nM T79062 CCN7R8 118728530 Ki = 2.99 nM T79062 C5O2NU 118729733 Ki = 17890 nM T79062 CB3Y2W 118731347 Ki = 116 nM T79062 CWZF06 118731348 Ki = 18 nM T79062 CA3O1H 118731349 Ki = 30 nM T79062 CU8P4W 118731350 Ki = 43 nM T79062 C8GKX6 118731351 Ki = 6 nM T79062 C2J4VC 118731352 Ki = 10 nM T79062 CF7NH5 118731353 Ki = 11 nM T79062 CQ8F6C 118731354 Ki = 77 nM T79062 CR9J0O 118731355 Ki = 135 nM T79062 CU12XM 118731356 Ki = 5 nM T79062 C4CEV7 118731357 Ki = 16 nM T79062 CU6T2D 118731358 Ki = 15 nM T79062 C95WKJ 118731359 Ki = 30 nM T79062 C20QAO 118731360 Ki = 40 nM T79062 CT6J8V 118731361 Ki = 22 nM T79062 C7QVJ4 118731362 Ki = 10 nM T79062 CA2X3O 118731363 Ki = 9 nM T79062 C4DV8I 118731364 Ki = 9 nM T79062 CHVY82 118731365 Ki = 12 nM T79062 CM5FG1 118731366 Ki = 9 nM T79062 C75OXS 118736395 Ki = 473 nM T79062 C74FCM 118736396 Ki = 61 nM T79062 C3F8PA 118736397 Ki > 1000 nM T79062 CHI8V7 121209051 Ki = 322 nM T79062 C7W3EY 122178698 Ki = 69 nM T79062 CF8P1H 122178699 Ki = 15 nM T79062 C48MFR 122178700 Ki = 24 nM T79062 CZ72QS 122178701 Ki = 58 nM T79062 C4VY8A 122178702 Ki = 52 nM T79062 C2KF4Z 122178703 Ki = 28 nM T79062 CX6MJ2 122178704 Ki = 34 nM T79062 CA53KF 122178705 Ki = 24 nM T79062 C8XD3F 122178706 Ki = 38 nM T79062 CTRC59 122178707 Ki = 22 nM T79062 C5QV8D 122178708 Ki = 50 nM T79062 C84UED 122178709 Ki = 20 nM T79062 CV96JK 122178710 Ki = 23 nM T79062 CM89KS 122178711 Ki = 54 nM T79062 C7ODW3 122195524 Ki > 900 nM T79062 CBHT01 122377930 Ki = 9 nM T79062 CG63UZ 122483217 Ki = 281.84 nM T79062 C3RX0B 122483224 Ki = 2336 nM T79062 C57RDF 122483225 Ki = 1071.52 nM T79062 C7PL6Q 122483228 Ki = 588.84 nM T79062 CW32JF 122483234 Ki = 251.19 nM T79062 C7K4ZC 122483237 Ki = 1307 nM T79062 C4JFD9 122483243 Ki = 549.54 nM T79062 CZ27HR 122483245 Ki = 151.36 nM T79062 C89LZM 122483248 Ki = 794.33 nM T79062 CM8HO9 122483250 Ki = 616 nM T79062 CB9U5S 122483253 Ki = 1398 nM T79062 CL4J6V 122483257 Ki = 831.76 nM T79062 C86NGA 122483259 Ki = 309.03 nM T79062 C24ZNM 122483261 Ki = 512.86 nM T79062 C2SWA8 122483263 Ki = 1047.13 nM T79062 C1G4YN 122483273 Ki = 676.08 nM T79062 CLW53P 122483274 Ki = 86 nM T79062 C8IZ9U 122483279 Ki = 949 nM T79062 CO63ET 122483280 Ki = 30 nM T79062 CJ84WM 122483287 Ki = 125.89 nM T79062 C5IV3P 122483288 Ki = 1281 nM T79062 C0Y7NI 122483295 Ki = 1905.46 nM T79062 CKSQ23 122483303 Ki = 2137.96 nM T79062 C4QM2E 124247485 Ki = 104 nM T79062 CLWM12 126720394 Ki = 8748 nM T79062 C8Q1JB 126720403 Ki = 11920 nM T79062 C1U3SZ 126720425 Ki = 7139 nM T79062 C5G8FD 126720440 Ki = 12340 nM T79062 CD50YM 127024949 Ki = 20 nM T79062 C4GF2D 127024950 Ki = 40 nM T79062 CJ76IB 127024951 Ki = 4 nM T79062 CKB42V 127025036 Ki = 157 nM T79062 CIHZ54 127025242 Ki = 2 nM T79062 CCY7P3 127025243 Ki = 1 nM T79062 CNJ4Z1 127025244 Ki = 9 nM T79062 CTBN56 127026052 Ki = 398.11 nM T79062 C26NMB 127026071 Ki = 74 nM T79062 C1YD7M 127026119 Ki = 344 nM T79062 CUO7Y8 127026120 Ki = 27 nM T79062 CDU21O 127026131 Ki = 4 nM T79062 C9HDP8 127026132 Ki = 70 nM T79062 CTYP30 127026133 Ki = 14 nM T79062 C19BOM 127026141 Ki = 50 nM T79062 CZFB49 127026142 Ki = 285 nM T79062 C2FT3B 127026143 Ki = 197 nM T79062 CP4J5H 127026144 Ki = 264 nM T79062 C6BIU4 127026145 Ki = 201 nM T79062 C1FA2U 127026146 Ki = 198 nM T79062 CE43NR 127026147 Ki = 39 nM T79062 CDAP16 127026434 Ki = 1918 nM T79062 C2XO3L 127026443 Ki = 54 nM T79062 C80QHX 127026444 Ki = 17 nM T79062 CBF64M 127026450 Ki = 12 nM T79062 CO1FB4 127026451 Ki = 14 nM T79062 CC13RA 127026452 Ki = 20 nM T79062 CBE56W 127026514 Ki = 74 nM T79062 C0SZI4 127026515 Ki = 38 nM T79062 CX6EI2 127026750 Ki = 19 nM T79062 CEG15O 127026751 Ki = 16 nM T79062 C1J4QY 127026752 Ki = 14 nM T79062 C0WB2U 127026753 Ki = 7 nM T79062 C62UMZ 127027143 Ki = 602.56 nM T79062 C4L0KU 127027144 Ki = 363.08 nM T79062 C0UOJ6 127027386 Ki = 72 nM T79062 C9IH1A 127027387 Ki = 26 nM T79062 C0TC7E 127027388 Ki = 53 nM T79062 CZ4W6I 127027389 Ki = 168 nM T79062 C4YR7A 127027390 Ki = 162 nM T79062 C3FA0I 127027391 Ki = 319 nM T79062 CC71UE 127027715 Ki = 292 nM T79062 CY2TW9 127028152 Ki = 223 nM T79062 CAZJ04 127028153 Ki = 89 nM T79062 CR48GO 127028154 Ki = 234 nM T79062 C8MC1I 127028408 Ki = 1023.29 nM T79062 CD8H7W 127028471 Ki = 47 nM T79062 C4EAY5 127028472 Ki = 10 nM T79062 CUS8R9 127028473 Ki = 14 nM T79062 CA10BY 127028634 Ki = 163 nM T79062 CZ26YR 127028797 Ki = 17 nM T79062 CI2R1N 127028798 Ki = 56 nM T79062 CS8GJ5 127028799 Ki = 837 nM T79062 CU0WQ3 127029375 Ki = 908 nM T79062 CS1GX5 127029649 Ki = 1190 nM T79062 C9N3BE 127029650 Ki = 141 nM T79062 CQFS48 127029651 Ki = 177 nM T79062 C7F3YE 127029652 Ki = 79 nM T79062 CZ61LK 127034966 EC50 > 5011.87 nM T79062 CA0SN5 127034967 EC50 > 5011.87 nM T79062 CQ0ZT9 127035062 Ki = 700 nM T79062 CU49VE 127036186 Ki = 154.88 nM T79062 CG06BD 127036932 Ki = 74.13 nM T79062 CVW71O 127036953 Ki = 48.98 nM T79062 C7N5DF 127037679 Ki = 8 nM T79062 CD13VY 127037680 Ki = 24 nM T79062 CTE43C 127037681 Ki = 19 nM T79062 C0LGK6 127037682 Ki = 21 nM T79062 C2XBE8 127037921 Ki = 49 nM T79062 CX0CN4 127037922 Ki = 18 nM T79062 CDAE15 127038033 Ki = 7 nM T79062 CFA6Q8 127038034 Ki = 44 nM T79062 CERL85 127038035 Ki = 49 nM T79062 C8TC9G 127038281 Ki = 10 nM T79062 CPK2Z7 127038282 Ki = 84 nM T79062 CYJ2D5 127039593 Ki = 56 nM T79062 CQED51 127039753 Ki = 7 nM T79062 CL4E2K 127039754 Ki = 36 nM T79062 CES26L 127039755 Ki = 6 nM T79062 CQ36LP 127039756 Ki = 7 nM T79062 C7KA2C 127040443 Ki = 200 nM T79062 CKBZ01 127040444 Ki = 42 nM T79062 CFAB12 127040760 Ki = 8 nM T79062 CWQ47G 127040761 Ki = 28 nM T79062 C8D4AV 127040908 Ki = 13 nM T79062 CE12AY 127041106 Ki = 19 nM T79062 C71LGS 127041107 Ki = 9 nM T79062 C6RI9V 127041108 Ki = 8 nM T79062 C15BGV 127041244 Ki = 9 nM T79062 CU0J4S 127041258 Ki = 18 nM T79062 C20MZH 127041259 Ki = 10 nM T79062 CP16CZ 127041260 Ki = 70 nM T79062 CZT53S 127041261 Ki = 68 nM T79062 C0FJP2 127041563 Ki = 58 nM T79062 CUC3F9 127041564 Ki = 58 nM T79062 COG9D2 127041874 Ki = 100 nM T79062 CS4WH1 127042184 Ki = 5 nM T79062 C13AIN 127042185 Ki = 7 nM T79062 CR59TP 127042539 Ki = 56 nM T79062 C54IZC 127042540 Ki = 28 nM T79062 C8G1HF 127042841 Ki = 53 nM T79062 CC7BU0 127049059 Ki = 1511 nM T79062 C42FHY 127049060 Ki > 10000 nM T79062 CF2QY9 127049061 Ki = 286 nM T79062 CX53AC 127050632 Ki = 1584.89 nM T79062 CTL0S1 127051516 Ki = 626 nM T79062 CTL8J1 127051843 Ki = 755 nM T79062 CF6V9Q 127051844 Ki = 12 nM T79062 C8TNB1 127051845 Ki = 16.98 nM T79062 C5ONG1 127051864 Ki = 1000 nM T79062 CVQW26 127051865 Ki = 79.43 nM T79062 CRF85X 127052458 Ki = 10 nM T79062 CCY71I 127052465 Ki = 330 nM T79062 C2E9VX 127052467 Ki = 51.29 nM T79062 CPO4C3 127052468 Ki = 86 nM T79062 CSQ2N8 127052486 Ki = 313 nM T79062 C4YJ8H 127052487 Ki = 111 nM T79062 CT9RS4 127052488 Ki = 778 nM T79062 CLU7C1 127052757 Ki = 26.92 nM T79062 C95KYT 127052758 Ki = 100 nM T79062 CYNR02 127052759 Ki = 48.98 nM T79062 C14YJU 127052778 Ki = 501.19 nM T79062 C1JAS7 127052779 Ki = 189 nM T79062 C7MQK8 127053042 Ki = 22.5 nM T79062 C50GOC 130442480 Ki = 8100 nM T79062 CM04RF 130442572 Ki = 4100 nM T79062 C4LJ2Y 132503215 Ki = 55 nM T79062 CM8B1L 132525569 Ki = 7.1 nM T79062 CU5L0K 132525570 Ki = 1.6 nM T79062 CA10SQ 132547275 Ki = 44.8 nM T79062 C6E1GN 132547276 Ki = 23.5 nM T79062 C6VTW3 132547277 Ki = 35.1 nM T79062 CI70OP 132547278 Ki = 45.1 nM T79062 C3Q1LA 132547279 Ki = 8.42 nM T79062 CAVB41 132584404 Ki > 10000 nM T79062 CS0MB3 132938109 Ki = 33 nM T79062 C8O2EP 134130246 Ki = 37 nM T79062 C8M9FH 134130379 Ki = 613 nM T79062 CA4GX3 134130447 Ki = 143 nM T79062 C7ZDA2 134130462 Ki = 53.7 nM T79062 CWL50Q 134130594 Ki = 1310 nM T79062 C8TG2O 134130846 Ki = 327 nM T79062 CHP3J4 134131015 Ki = 1377 nM T79062 CQ4IF8 134131147 Ki = 94.7 nM T79062 C6N5FS 134131151 Ki = 1328 nM T79062 CH4XB2 134131159 Ki = 990 nM T79062 CR32SP 134131265 Ki = 181 nM T79062 C0JKL5 134131283 Ki = 276 nM T79062 C0RQC6 134131976 Ki = 27 nM T79062 CQX4U3 134133064 Ki = 6.31 nM T79062 CTS3J4 134133483 Ki = 18.5 nM T79062 C0J2ML 134133604 Ki = 0.4677 nM T79062 CP0E5M 134133632 Ki = 497 nM T79062 CM0TS6 134133967 Ki = 44.67 nM T79062 CNV91Q 134134210 Ki = 23 nM T79062 C0ZLJ3 134134279 Ki = 648 nM T79062 CC1DO8 134134456 Ki = 25.5 nM T79062 CMS79H 134135372 Ki = 1038 nM T79062 C2Q3JY 134135516 Ki = 76 nM T79062 CJG3U0 134136134 Ki = 9.5 nM T79062 CGX03A 134136246 Ki = 131.83 nM T79062 C4VR6O 134137104 Ki = 18 nM T79062 C08ZBY 134137332 Ki = 32 nM T79062 CXF52V 134137560 Ki = 15.5 nM T79062 CN4LI8 134137732 Ki = 11.5 nM T79062 CWO5R6 134138168 Ki = 18 nM T79062 CRC2V0 134139826 Ki = 54 nM T79062 CG30KH 134140472 Ki = 126 nM T79062 CHK39T 134141166 Ki = 8 nM T79062 CLW86T 134141354 Ki = 257 nM T79062 C2NOX7 134141985 Ki = 34 nM T79062 CK54QW 134142259 Ki = 259 nM T79062 C6PSI9 134142907 Ki = 87 nM T79062 CR5L4K 134144303 Ki = 138 nM T79062 CYF16Z 134144798 Ki = 3063 nM T79062 C80TGJ 134144864 Ki = 25 nM T79062 CGW1D0 134145143 Ki = 1476 nM T79062 CK5RU9 134145903 Ki = 10 nM T79062 C2E0ID 134146185 Ki = 44 nM T79062 CC9P2T 134146194 Ki = 43.65 nM T79062 CV0QZ5 134147124 Ki = 52 nM T79062 C41XSD 134147935 Ki = 108 nM T79062 CFD13P 134147951 Ki = 1019 nM T79062 C8NBO0 134148917 Ki = 772 nM T79062 CBU81N 134149168 Ki > 10000 nM T79062 C0J8HT 134150597 Ki = 691 nM T79062 CE6LN3 134151118 Ki = 21 nM T79062 CLU34D 134151427 Ki = 265 nM T79062 C2JN8Y 134151729 Ki = 36.5 nM T79062 C76BZW 134151980 Ki = 16 nM T79062 CIV4H5 134152583 Ki = 254 nM T79062 CB6M5Y 134153538 Ki = 144 nM T79062 CX4W7F 134153716 Ki = 12 nM T79062 C79TEI 134154068 Ki = 25 nM T79062 C5B4GR 134154108 Ki = 1123 nM T79062 CMJ1U3 134154387 Ki = 65 nM T79062 C4M0FW 134154531 Ki = 79 nM T79062 C4VGJ5 134154679 Ki = 67 nM T79062 C6QAY2 134155116 Ki = 1.585 nM T79062 C79QLN 134155460 Ki = 91 nM T79062 CIUZ94 134155476 Ki = 10.5 nM T79062 C90QNV 134155645 Ki = 14 nM T79062 C97EWM 134155651 Ki = 389 nM T79062 CVR87Q 134156222 Ki = 125.89 nM T79062 CAB4K6 134156305 Ki = 19 nM T79062 C50XNE 134156520 Ki = 4.5 nM T79062 CUHE07 134157171 Ki = 6.5 nM T79062 CV8JU6 134157289 Ki = 73 nM T79062 CL6DN0 134157769 Ki = 14.5 nM T79062 C5IM7X 135367399 Ki = 363.08 nM T79062 C41JQV 135367400 Ki = 501.19 nM T79062 C2RN9U 135367403 Ki = 1407 nM T79062 C74JIA 135367404 Ki = 881 nM T79062 C6N8GM 135367405 Ki = 46.77 nM T79062 C6LU0C 135367816 Ki = 70 nM T79062 CTX68N 135367817 Ki = 883 nM T79062 CD2TH9 135367820 Ki = 52.48 nM T79062 CM7SA8 135367821 Ki = 369 nM T79062 CP21LA 135367855 Ki = 425 nM T79062 C5AMD9 135367857 Ki = 16 nM T79062 C6SKM3 135367858 Ki = 707.95 nM T79062 C5URG0 135367869 Ki = 1230.27 nM T79062 CBA7P6 135367917 Ki = 1436 nM T79062 C9DVI7 135367936 Ki = 386 nM T79062 CR0U6A 135367959 Ki = 316.23 nM T79062 CVE08Y 135458392 Ki = 15.3 nM T79062 CP7HN4 135458393 Ki = 33.3 nM T79062 CS8XJ6 135458394 Ki = 13.2 nM T79062 C9B7XA 135458410 Ki = 23.3 nM T79062 CFV9A3 135458427 Ki = 4.2 nM T79062 CKX4N8 135458428 Ki = 38.9 nM T79062 C9ZCL5 135458672 Ki = 4194 nM T79062 CTE23K 135464118 Ki = 512 nM T79062 CD6L8Q 135895192 Ki = 13.6 nM T79062 CA1M8B 135966709 Ki = 2.4 nM T79062 CUKO20 136020617 Ki > 10000 nM T79062 COF0U5 136020618 Ki > 10 nM T79062 CF89JI 136030596 Ki > 10000 nM T79062 CE8GB9 136030693 Ki > 10000 nM T79062 C65VFI 136030744 Ki > 10000 nM T79062 COIX80 136054961 Ki > 10000 nM T79062 C19GLK 136116062 Ki = 366.3 nM T79062 CQ2GP6 136118614 Ki = 1223 nM T79062 C8RH6M 136118617 Ki = 4114 nM T79062 CG5TX8 136118653 Ki = 3350 nM T79062 C40LYH 136118659 Ki = 5367 nM T79062 CY5GU4 136118730 Ki = 799 nM T79062 CB12QP 136152964 Ki = 24.8 nM T79062 CFX06E 136152966 Ki = 17.6 nM T79062 C37YXA 136152971 Ki = 7.7 nM T79062 CY0C1X 136152972 Ki = 1704 nM T79062 CX53NC 136180316 Ki = 145 nM T79062 CZ7WT9 136180317 Ki = 21.2 nM T79062 CQP2Y6 136180318 Ki = 1135 nM T79062 CQT9H5 136180319 Ki = 228 nM T79062 CLPU18 136180320 Ki = 11.9 nM T79062 C0LO6Q 136180321 Ki = 101 nM T79062 CAE39V 136188797 Ki > 10000 nM T79062 CWP0V5 136216703 Ki = 1600 nM T79062 CLAP52 136259032 Ki > 10000 nM T79062 CHM36P 137631892 Ki = 52 nM T79062 CU01TV 137633827 Ki > 10000 nM T79062 CC51JN 137635185 Ki > 10000 nM T79062 C94VXJ 137635884 Ki = 95 nM T79062 CFM92C 137636384 Ki = 3692 nM T79062 CDX39B 137637994 Ki = 142 nM T79062 C3LYX9 137641832 Ki > 10000 nM T79062 C5WS6Q 137642134 Ki = 14 nM T79062 CWUM83 137644521 Ki > 10000 nM T79062 CDA80E 137644790 Ki = 36 nM T79062 CZ8CU6 137645501 Ki = 56 nM T79062 CCP38D 137645926 Ki = 37 nM T79062 CVX74E 137646045 Ki = 438 nM T79062 CPI68E 137646281 Ki = 128 nM T79062 CMXI62 137649997 Ki = 209 nM T79062 C52IRM 137650705 Ki = 37 nM T79062 CKG08R 137650961 Ki = 165 nM T79062 CU4S1W 137651887 Ki = 5 nM T79062 CVK26R 137652044 Ki = 174 nM T79062 CHFK13 137652210 Ki > 10000 nM T79062 C51CGJ 137652310 Ki = 29 nM T79062 C2E3FV 137653850 Ki = 18 nM T79062 CX82HS 137654666 Ki = 32 nM T79062 C0SKV1 137654850 Ki > 10000 nM T79062 C4VG0U 137655411 Ki = 39 nM T79062 CO3L7F 137656918 Ki > 10000 nM T79062 CX4D7Y 137660741 Ki = 52 nM T79062 C0R6XM 138691314 Ki = 6 nM T79062 CU3Y7W 138691316 Ki = 20 nM T79062 CH2W4P 138691317 Ki = 531 nM T79062 CHSC40 138691321 Ki = 36 nM T79062 C18UZA 138691329 Ki = 42 nM T79062 C1XWV0 138691338 Ki = 30 nM T79062 C6LE1A 138691362 Ki = 44 nM T79062 CN9R4A 138691364 Ki = 5 nM T79062 C8H2KR 138691366 Ki = 302 nM T79062 C2Z9CD 139488518 Ki = 386 nM T79062 CJK95T 139488527 Ki = 22 nM T79062 CZ6H9M 139488539 Ki = 16 nM T79062 CAF2H8 139488606 Ki = 4 nM T79062 C54CIL 139488740 Ki = 18 nM T79062 CN3G0A 140936451 Ki > 10000 nM T79062 C4EU2S 141745651 Ki = 0.99 nM T79062 CCO6R0 141745657 Ki = 2.2 nM T79062 CO5DR9 145949220 Ki = 23 nM T79062 CWAF96 145949371 Ki = 10 nM T79062 CHG2W6 145950605 Ki = 9 nM T79062 COU57L 145950881 Ki = 7 nM T79062 CD4M6B 145951915 Ki = 85 nM T79062 C78AUI 145952711 Ki = 8 nM T79062 CA2J5S 145954503 Ki = 71200 nM T79062 C0JO8B 145954831 Ki = 10 nM T79062 CHI1V8 145956064 Ki = 566 nM T79062 CSER68 145956892 Ki = 20 nM T79062 CLVI07 145957637 Ki = 213 nM T79062 C91IDE 145958490 Ki = 1205 nM T79062 C8VS7K 145959257 Ki = 94 nM T79062 CSIZ31 145959706 Ki = 12 nM T79062 C67GQI 145961372 Ki = 2797 nM T79062 C4Y1PK 145963314 Ki = 6 nM T79062 C7KC3T 145963830 Ki > 10000 nM T79062 C5VWM7 145963860 Ki = 74 nM T79062 CCK5G1 145963863 Ki = 902 nM T79062 C4Y2AL 145964000 Ki = 3142 nM T79062 CV7YW9 145964086 Ki = 170 nM T79062 CHDN35 145964150 Ki > 10000 nM T79062 CR2B9G 145964154 Ki = 290 nM T79062 C1KH2E 145964159 Ki = 3600 nM T79062 C7YKQ4 145964390 Ki = 93 nM T79062 C95NZO 145964427 Ki = 89 nM T79062 C2P5NK 145964621 Ki = 67 nM T79062 CK0T1M 145964694 Ki = 213 nM T79062 C6T4RY 145964846 Ki = 90 nM T79062 CE9K3L 145964944 Ki = 12 nM T79062 C12OVL 145965034 Ki > 10000 nM T79062 CBS74V 145965054 Ki = 4 nM T79062 C9D8IB 145965203 Ki = 15 nM T79062 C1MIR9 145965401 Ki = 258 nM T79062 CLP94W 145965668 Ki = 245 nM T79062 C8TF9G 145965840 Ki = 121 nM T79062 C5W4LM 145965940 Ki > 10000 nM T79062 C53EFW 145966154 Ki = 547 nM T79062 CB05QA 145966199 Ki = 59 nM T79062 C1T4DN 145966418 Ki = 55 nM T79062 CV03XA 145967457 Ki = 1580 nM T79062 C81VUO 145967771 Ki > 10 nM T79062 CJS56K 145967795 Ki > 10000 nM T79062 CQ8EM6 145969402 Ki = 29 nM T79062 CA82FL 145970078 Ki = 2 nM T79062 CF74MR 145971390 Ki = 1671 nM T79062 C1T7GL 145971527 Ki = 12500 nM T79062 C8A2XG 145971561 Ki = 38 nM T79062 CN64ZR 145971588 Ki = 1154 nM T79062 CQJ5O8 145971635 Ki > 10000 nM T79062 C56RAO 145972025 Ki = 284 nM T79062 C79TNE 145972796 Ki > 10000 nM T79062 CJHI43 145972875 Ki = 52 nM T79062 CS7WG8 145973438 Ki = 1154 nM T79062 C8KYV6 145973487 Ki = 313 nM T79062 CEOY46 145973577 Ki = 388 nM T79062 CL74IP 145973853 Ki = 6 nM T79062 CR0CX6 145974087 Ki = 50 nM T79062 C6XIN0 145974114 Ki > 10000 nM T79062 C8KZ5T 145974165 Ki = 0.75 nM T79062 C05IVJ 145974184 Ki = 172 nM T79062 CW6EX3 145974189 Ki = 32 nM T79062 CD8ZL6 145974750 Ki > 10 nM T79062 C3WG0J 145975106 Ki = 52 nM T79062 C6PH4F 145975226 Ki > 10000 nM T79062 CN8U3P 145975289 Ki = 86 nM T79062 CSVR94 145975713 Ki = 408 nM T79062 COY2P3 145975720 Ki = 21 nM T79062 CL7EX5 145975776 Ki = 1050 nM T79062 C1BI8E 145975778 Ki = 534 nM T79062 C7R2MD 145975905 Ki = 100 nM T79062 C71CYU 145975946 Ki > 10000 nM T79062 C0V4AL 145975992 Ki = 275 nM T79062 C2TN8W 145976085 IC50 > 10000 nM T79062 C8XFM7 145976120 Ki = 3027 nM T79062 CF5B0W 145976158 Ki = 41 nM T79062 C8BJI2 145976292 Ki = 58 nM T79062 CZ5XK2 145976408 Ki = 67 nM T79062 C14OJW 145976618 Ki = 34 nM T79062 C0LRB2 145976686 Ki = 110 nM T79062 C34XME 145976696 Ki = 70 nM T79062 CTCM92 145976698 Ki = 415 nM T79062 CIZ69S 145976722 Ki = 228 nM T79062 CT7WO5 145976787 Ki = 213 nM T79062 CI8AN3 145976890 Ki = 32 nM T79062 C81CSM 145976946 Ki = 931 nM T79062 CXDR94 145977222 Ki = 3160 nM T79062 C8NW7Y 145977256 Ki = 43 nM T79062 CHS96B 145977297 Ki = 3.2 nM T79062 C6BFY7 145977338 Ki = 7400 nM T79062 C4L8EZ 145977467 Ki = 64 nM T79062 CC1DZ5 145977555 Ki = 204 nM T79062 C0Y6QO 145977799 Ki = 3300 nM T79062 C3BI1R 145978113 Ki > 10000 nM T79062 CP8C6M 145978146 Ki = 104 nM T79062 C6HQI0 145978420 Ki = 203 nM T79062 C8VL3Y 145978472 Ki = 529 nM T79062 C82NXP 145978482 Ki = 602 nM T79062 CQU8R0 145978665 Ki > 10000 nM T79062 C6AV9G 145978819 Ki > 10000 nM T79062 C20XQJ 145979626 Ki = 3609 nM T79062 C87MSW 145980271 Ki = 812 nM T79062 CW2CO4 145980458 Ki = 11 nM T79062 C8I7QL 145980875 Ki = 1120 nM T79062 CPK34X 145981875 Ki = 1.1 nM T79062 COY79P 145982165 Ki = 5 nM T79062 CEK60A 145982506 Ki = 165 nM T79062 CI59TX 145983018 Ki = 1119 nM T79062 CYC58R 145983059 Ki = 45 nM T79062 C4F5OT 145983128 Ki = 14 nM T79062 C5ZG9M 145983139 Ki = 7 nM T79062 CV2GU9 145983144 Ki = 65 nM T79062 C4PKM2 145983390 Ki = 19 nM T79062 C9LR8C 145983405 Ki = 0.55 nM T79062 CIAF74 145983468 Ki = 57 nM T79062 CE7MF4 145983751 Ki = 69 nM T79062 CDQ4U7 145983760 Ki = 19 nM T79062 CYW9B2 145983794 Ki = 32 nM T79062 C8I1WG 145983961 Ki = 3 nM T79062 CP5H4D 145984065 Ki = 8 nM T79062 CJ35DM 145984299 Ki = 9 nM T79062 CU7E4M 145984511 Ki = 51 nM T79062 C6JUY0 145984737 Ki = 12 nM T79062 CID02G 145984807 Ki = 672 nM T79062 CM5X3V 145985050 Ki = 0.4 nM T79062 CG10LK 145985224 Ki = 17 nM T79062 CFJ9B3 145985233 Ki = 12 nM T79062 C5AOI6 145985289 Ki = 24 nM T79062 CW30NA 145985505 Ki = 10 nM T79062 C7ZRP1 145985527 Ki = 12 nM T79062 C2XY8Q 145985533 Ki = 7 nM T79062 C7NI4X 145985585 Ki = 6 nM T79062 C9LJ5T 145985692 Ki = 1 nM T79062 C7QIX0 145985718 Ki = 52 nM T79062 C6V5QS 145985823 Ki = 12 nM T79062 C07GKD 145985958 Ki = 1340 nM T79062 CCM18E 145986031 Ki = 22 nM T79062 CR0XQ3 145986138 Ki = 31 nM T79062 CT37DW 145986720 Ki = 824 nM T79062 CNJH37 145986752 Ki = 949 nM T79062 C3VN5O 145987559 Ki = 165 nM T79062 CI0PA9 145987771 Ki = 3.3 nM T79062 CIS9P2 145988193 Ki = 12 nM T79062 CUGO10 145988693 Ki = 1574 nM T79062 C9D2OG 145988738 Ki = 3 nM T79062 C4C0YP 145988913 Ki = 172 nM T79062 CDY48U 145989143 Ki = 0.26 nM T79062 C3GPR9 145990093 Ki = 2085 nM T79062 C2Q5UK 145990353 Ki = 3 nM T79062 CT7AB8 145990459 Ki = 2172 nM T79062 C4GV8Q 145990586 Ki = 120 nM T79062 CVBR36 145991084 Ki = 0.79 nM T79062 C9TK6G 145991864 Ki = 2.6 nM T79062 CB8CM6 145992305 Ki = 209 nM T79062 CCP2U1 145992489 Ki = 10000 nM T79062 CLPU06 145992567 Ki = 224 nM T79062 CBI94R 145992877 Ki = 1.1 nM T79062 CI19KS 145993474 Ki = 2.3 nM T79062 C0TL8E 145993714 Ki = 19 nM T79062 CC2G1V 146025727 Ki = 3800 nM T79062 C5ZOJ3 146680920 Ki = 7832 nM T79062 CG97ER 146709966 Ki = 1000 nM T79062 CF5B2L 147653864 Ki = 398.11 nM T79062 C9T0PS 153061504 Ki = 691.83 nM T79062 CAF36V 153287539 Ki = 1000 nM T79062 C1FA0K 153287541 Ki = 19.95 nM T79062 CEQ69Z 153287542 Ki = 23.44 nM T79062 C6P3SR 153287553 Ki = 6.3 nM T79062 C3G5CJ 153287557 Ki = 199.53 nM T79062 CW31CT 153287566 Ki = 2.692 nM T79062 CYP86E 153287567 Ki = 199.53 nM T79062 CS73ZC 153287568 Ki = 1258.93 nM T79062 CV9G7Z 153287572 Ki > 10000 nM T79062 CO85KL 153287574 Ki = 1000 nM T79062 CZ1K4D 155510674 Ki = 21 nM T79062 CLX3D8 155510732 IC50 = 650 nM T79062 CC3KP7 155510927 Ki = 1148 nM T79062 CM4RB0 155511262 Ki = 3147 nM T79062 C9KX6O 155511928 Ki = 280 nM T79062 CZ7HP4 155512406 Ki = 40.1 nM T79062 C4OL0A 155512409 Ki = 3.43 nM T79062 CXF90M 155512487 Ki = 895 nM T79062 CO68LC 155512944 Ki = 49 nM T79062 C90FST 155513438 Ki = 51 nM T79062 C95QOT 155514378 Ki = 2352 nM T79062 C3SQI7 155514459 Ki > 10000 nM T79062 CI4DT8 155514575 Ki = 2455 nM T79062 CJUI87 155514774 Ki = 45 nM T79062 CQ84DA 155514889 Ki = 298 nM T79062 C3NB0D 155515324 Ki = 98430 nM T79062 C0Q8PR 155515407 Ki = 1833 nM T79062 CWO56B 155515415 Ki > 10000 nM T79062 CU0PY6 155515687 Ki = 9.42 nM T79062 C2TN5D 155515890 Ki = 184 nM T79062 C7KT0D 155515919 Ki = 1096 nM T79062 C13LOV 155515942 Ki = 6660 nM T79062 C7OF4C 155516118 Ki = 13750 nM T79062 CJ1Z0D 155516162 Ki > 10000 nM T79062 CG5M1O 155516282 Ki = 3743 nM T79062 CG53LH 155516399 Ki = 0.85 nM T79062 CU8TC0 155517162 Ki = 25 nM T79062 CW0B5K 155518159 Ki > 10000 nM T79062 CYB12O 155518974 Ki = 116500 nM T79062 CHVF41 155519045 Ki = 401 nM T79062 CCEZ93 155519102 Ki = 38730 nM T79062 CQD2J7 155519393 Ki = 9855 nM T79062 C2SXT1 155519515 Ki = 167 nM T79062 C0KLD8 155519559 Ki = 6248 nM T79062 C07BTO 155519598 Ki = 291 nM T79062 CUSA24 155519891 Ki = 1258.93 nM T79062 C5FL7R 155520499 Ki = 822 nM T79062 C8OC3W 155520552 Ki = 140 nM T79062 CTV2F6 155521010 Ki = 380 nM T79062 CQ76MP 155521503 Ki = 3715 nM T79062 C1OS6D 155522116 Ki > 10000 nM T79062 C98RDQ 155522218 Ki = 1115 nM T79062 C2TV4Y 155522487 Ki > 10000 nM T79062 CP6H1D 155522562 Ki = 432 nM T79062 CUQ61M 155522867 Ki = 7.54 nM T79062 CUG8L3 155522920 Ki > 10000 nM T79062 CD9QU6 155523519 Ki = 20 nM T79062 C5KYB4 155524228 Ki = 458 nM T79062 C6APG2 155524374 Ki = 36.6 nM T79062 CK4B0R 155524491 Ki = 1361 nM T79062 CUO93F 155524808 Ki = 305 nM T79062 CQB0M8 155524884 Ki > 10000 nM T79062 C65UZD 155524956 Ki = 286 nM T79062 C6MZJ9 155525703 Ki = 74 nM T79062 C81OCJ 155526014 Ki = 80.3 nM T79062 CZ81JA 155526026 Ki = 120 nM T79062 C1U2XO 155526651 Ki = 119 nM T79062 CXH79K 155526720 Ki = 11 nM T79062 CW68KC 155528355 Ki > 10000 nM T79062 C7C1EF 155528967 Ki = 1444 nM T79062 C5J7AU 155529153 Ki = 4247 nM T79062 C9KS5C 155529450 Ki = 58 nM T79062 CKZ25Y 155529679 Ki = 195 nM T79062 C3X4IA 155530328 Ki = 233 nM T79062 C9PC3D 155530350 Ki = 5996 nM T79062 CVLC03 155530779 Ki = 871 nM T79062 C98YQF 155531012 Ki = 258 nM T79062 C4W6VC 155531065 Ki = 1622 nM T79062 C5HWP4 155531362 Ki > 10000 nM T79062 CKDE38 155531753 Ki = 1 nM T79062 CCT8V9 155531846 Ki = 9531 nM T79062 C05KFL 155532137 Ki = 56.2 nM T79062 CMPU81 155532470 Ki > 10000 nM T79062 CX35QS 155532545 Ki > 10000 nM T79062 CX6DV4 155533028 Ki = 696 nM T79062 C23GDV 155533534 Ki = 1712 nM T79062 C3OEH2 155533648 Ki = 710 nM T79062 C15RYP 155533660 Ki > 10000 nM T79062 CY01GZ 155533850 Ki = 1384 nM T79062 CP3J8B 155534152 Ki = 3467 nM T79062 C3L0CP 155534184 Ki = 2431 nM T79062 CG85SB 155534301 Ki = 475 nM T79062 CG8Y7W 155534312 Ki = 366 nM T79062 C3VGT0 155534362 Ki = 1922 nM T79062 CW7SV9 155534575 Ki = 35 nM T79062 C75FSY 155534794 Ki = 2512 nM T79062 CTO4S9 155534839 Ki = 2 nM T79062 C6KF4E 155535154 Ki = 546 nM T79062 C8G7AW 155535428 Ki > 10000 nM T79062 C8O4IQ 155535827 Ki = 35 nM T79062 C14JEX 155535878 Ki = 776 nM T79062 CB79ZW 155536080 Ki > 10000 nM T79062 C5I1JA 155536087 Ki = 322 nM T79062 C72FLG 155536152 Ki = 3804 nM T79062 CW2SC8 155536533 Ki = 106 nM T79062 CTB93R 155536809 Ki = 462 nM T79062 C7FVE8 155537034 Ki = 6 nM T79062 C36FRH 155537074 Ki = 2095 nM T79062 CD75GP 155537227 Ki > 10000 nM T79062 CVS04L 155537788 Ki = 23 nM T79062 CB8IC7 155538144 Ki = 273 nM T79062 C5F2GI 155538236 Ki = 1092 nM T79062 COYG20 155538350 Ki = 933 nM T79062 C9TIU2 155538367 Ki = 53 nM T79062 CYC1P3 155538451 Ki = 73 nM T79062 CM08NT 155538716 Ki > 10000 nM T79062 CQ69UA 155538814 Ki = 5818 nM T79062 C0Q5NT 155538877 Ki = 133 nM T79062 CAT98F 155539483 Ki = 1158 nM T79062 C6S8BA 155539600 Ki = 4570 nM T79062 C9S2IA 155539605 Ki = 2765 nM T79062 C42GUK 155540147 Ki > 10000 nM T79062 C1X0IO 155540198 Ki = 197 nM T79062 C9J3BQ 155540635 Ki = 65.1 nM T79062 C1KA8C 155540755 Ki = 43.8 nM T79062 CR2K1T 155540795 Ki > 10000 nM T79062 CNU92V 155540807 Ki = 25 nM T79062 CUY87S 155540823 Ki = 119 nM T79062 COS2E7 155541072 Ki = 6417 nM T79062 CP7UG2 155541866 Ki = 3298 nM T79062 COZ46W 155541871 Ki = 53 nM T79062 CB62ZS 155542237 Ki = 2455 nM T79062 CXCW81 155542321 Ki = 11950 nM T79062 C9FS3Y 155542461 Ki > 10000 nM T79062 C9RV7W 155542678 Ki = 1.99 nM T79062 CT6HY4 155543250 Ki = 29 nM T79062 C68MSK 155543653 Ki = 8361 nM T79062 CZ7O0A 155544139 Ki = 5840 nM T79062 CD84VK 155544810 Ki = 336 nM T79062 C2XZD8 155545087 Ki = 404 nM T79062 CCX6T2 155545402 Ki = 3.3 nM T79062 CO9X1Z 155545526 Ki > 10000 nM T79062 CI0YL8 155545625 Ki = 70 nM T79062 C74GFO 155546189 Ki = 203 nM T79062 CH3W9N 155546350 Ki = 1445 nM T79062 C4UT5Z 155546595 Ki = 125 nM T79062 C98AIL 155546781 Ki = 3.54 nM T79062 CD02EN 155547436 Ki = 371 nM T79062 COJ27N 155547693 Ki = 10660 nM T79062 CAT9X4 155548275 Ki = 8511 nM T79062 C5LYE8 155548677 Ki = 5316 nM T79062 C0KZB5 155549018 Ki = 50.2 nM T79062 C87JGN 155549153 Ki > 10000 nM T79062 CGP8O5 155549315 Ki = 291 nM T79062 C52FRY 155549978 Ki = 192 nM T79062 C8HPN7 155551113 Ki = 420 nM T79062 C61IVC 155551353 Ki = 8 nM T79062 CHS71N 155551685 Ki = 119 nM T79062 CM26AV 155551704 Ki > 1000 nM T79062 C6E9LK 155552054 Ki = 366 nM T79062 CQ48CS 155552188 Ki = 0.9 nM T79062 CA1WS9 155552212 Ki = 5095 nM T79062 C38YJB 155552311 Ki = 2761 nM T79062 C87PTM 155552707 Ki = 11 nM T79062 CDQ7C2 155552798 Ki = 48960 nM T79062 CPV35U 155552826 Ki = 161 nM T79062 CDV6B9 155554036 Ki = 9247 nM T79062 CKF75H 155554324 Ki = 124 nM T79062 C6ZSU3 155554462 Ki = 2871 nM T79062 C8JKT1 155555378 Ki = 19.3 nM T79062 C2E5TR 155555506 Ki = 525 nM T79062 CUNK28 155555525 Ki > 10000 nM T79062 CO52HW 155556527 Ki = 5888 nM T79062 C1N5VF 155556756 Ki > 10000 nM T79062 CJCL47 155556806 Ki = 75.8 nM T79062 CJBX01 155557042 Ki = 199.53 nM T79062 C5QYS0 155557134 Ki = 34 nM T79062 CD2L3K 155557443 Ki = 21 nM T79062 CER48T 155557500 Ki > 10000 nM T79062 C2L0PC 155557720 Ki = 16 nM T79062 CF6H3V 155558408 Ki = 15180 nM T79062 C4I2OY 155558563 Ki = 27.8 nM T79062 C9TB5D 155559092 Ki = 2366 nM T79062 CP4JO7 155559794 Ki > 10000 nM T79062 COG70U 155560942 Ki = 7079 nM T79062 C2HF6P 155561581 Ki = 2329 nM T79062 COL7N8 155561901 Ki = 46 nM T79062 CL45NV 155561914 Ki = 17780 nM T79062 CJ57BI 155561978 Ki = 22 nM T79062 C0SDZ8 155561990 IC50 = 12 nM T79062 CW7M1D 155561995 Ki = 1112 nM T79062 C93KWN 155562202 Ki = 266 nM T79062 CO3C6L 155562423 Ki > 10000 nM T79062 C5AI0S 155562519 Ki = 641 nM T79062 C5BQ8U 155562652 Ki = 958 nM T79062 CF6B4W 155562834 Ki = 344 nM T79062 CZ6IA2 155562918 Ki = 514 nM T79062 CRCW25 155562997 Ki = 50 nM T79062 CBH14K 155563164 Ki > 10000 nM T79062 CG1L8E 155563286 Ki > 10000 nM T79062 C38WXS 155563374 Ki = 7322 nM T79062 C0INS4 155563826 Ki > 10000 nM T79062 CK0IW3 155563911 Ki = 6 nM T79062 C5TS7Q 155564824 Ki = 710 nM T79062 CQK8E3 155565209 Ki = 54.7 nM T79062 CE2YG1 155565215 Ki = 12.2 nM T79062 C2MIU5 155565813 Ki = 2730 nM T79062 C7P5VG 155566191 Ki = 206 nM T79062 C7O6YP 155566439 Ki = 16050 nM T79062 CG35LB 155566508 Ki = 24.2 nM T79062 CU46EB 155566665 Ki > 10000 nM T79062 C67LAG 155566854 Ki = 9120 nM T79062 CW1TN7 155566925 Ki = 14 nM T79062 C41UWT 155567307 Ki = 84 nM T79062 CA8OE0 155567476 Ki = 9.08 nM T79062 CC06FO 155567938 Ki = 1.86 nM T79062 CA68TK 155568224 Ki = 614 nM T79062 C4EX7C 155568246 Ki = 320 nM T79062 C4POS3 155568373 Ki = 32.7 nM T79062 C67MIN 155568606 Ki = 0.8 nM T79062 CXP3E4 155568794 Ki = 1501 nM T79062 CB5IP9 155569021 Ki = 166 nM T79062 C0CZK6 155569337 Ki > 10000 nM T79062 CP9V7M 155569396 Ki = 138 nM T79062 C3ZNX6 155569414 Ki = 552 nM T79062 CZ8RV4 155569568 Ki = 2170 nM T79062 C3N9VU 10251906 Ki > 500 nM T79062 CP9TR0 10324985 Ki = 9.1 nM T79062 D00CRA 1574 Ki = 1258 nM T79062 D00GSD 25107716 Ki = 0.58 nM T79062 D00MXS 5281703 IC50 > 350000 nM T79062 D00OBS 44559159 Ki > 10000 nM T79062 D00VRV 10171 Ki = 10 nM T79062 D00YEV 5281605 IC50 > 350000 nM T79062 D01KAX 135453290 EC50 = 5600 nM T79062 D01KVG 9843179 Ki = 1.995 nM T79062 D01WWC 16573 Ki = 20 nM T79062 D02HZG 888311 Ki = 2663 nM T79062 D02RAY 16754 Ki = 43 nM T79062 D02UWB 1809 Ki = 0.3981 nM T79062 D02YSX 197033 Ki = 7.943 nM T79062 D03DET 10287730 Ki = 501.19 nM T79062 D03NBX 637308 IC50 = 47600 nM T79062 D03TDN 1342 Ki = 83 nM T79062 D03TSY 24825775 Ki = 2.5 nM T79062 D03ZHB 44455973 Ki = 97.4 nM T79062 D04AQE 1833 Ki = 2 nM T79062 D04TPO 16006492 Ki = 15.85 nM T79062 D05EQG 5265 Ki = 19.95 nM T79062 D05GDP 599482 Ki = 1400 nM T79062 D05LKO 44414722 Ki = 840 nM T79062 D05XGR 6918647 Ki = 2511.89 nM T79062 D05ZUX 44207909 Ki >= 1000 nM T79062 D06VDN 443391 IC50 > 1000 nM T79062 D07JRV 46233381 Ki = 553 nM T79062 D07JTZ 9843889 Ki = 89 nM T79062 D07LRJ 5312149 Ki = 260 nM T79062 D08BCF 5011 Ki = 3033 nM T79062 D08CKM 9863250 Ki = 3 nM T79062 D08DOG 25130235 Ki = 5900 nM T79062 D08OFG 11177588 Ki > 10000 nM T79062 D08UOX 5281148 IC50 = 117500 nM T79062 D08VGJ 9904281 Ki = 294 nM T79062 D09BNS 439280 Ki = 2.12 nM T79062 D09RPR 16737207 Ki > 10000 nM T79062 D09RXU 45488131 Ki > 500 nM T79062 D09WIL 10028436 Ki = 1.995 nM T79062 D0B9TN 46233353 Ki = 4110 nM T79062 D0BG5H 11957684 Ki = 1.259 nM T79062 D0C5GF 6918515 Ki = 155 nM T79062 D0C5XQ 1832 Ki = 30 nM T79062 D0CA9H 25107518 Ki = 16.6 nM T79062 D0CK9K 6918513 Ki = 300 nM T79062 D0F0IA 11301655 Ki > 2000 nM T79062 D0F6CD 5202 Ki = 0.11 nM T79062 D0FF6S 16038374 IC50 > 10000 nM T79062 D0FU5E 10220053 Ki > 1000 nM T79062 D0G7QT 10131112 IC50 = 3000 nM T79062 D0G8CV 9954003 Ki = 7.943 nM T79062 D0H3KU 172267 Ki = 466 nM T79062 D0H7PC 6918553 Ki > 10000 nM T79062 D0H9QG 5312148 Ki = 31.6 nM T79062 D0HE4S 68788 Ki = 18 nM T79062 D0I0ML 35985234 Ki = 7.5 nM T79062 D0J6JT 1355 Ki = 304 nM T79062 D0K0HU 16747715 Ki = 7.6 nM T79062 D0K5NZ 68848 Ki = 7.943 nM T79062 D0KS0I 24894910 EC50 > 10000 nM T79062 D0L5MW 181743 Ki = 67 nM T79062 D0LT5D 11267988 Ki = 3.38 nM T79062 D0LV7U 10667433 Ki = 32 nM T79062 D0O3GF 1220 Ki = 388 nM T79062 D0OG0R 10337743 IC50 = 4764 nM T79062 D0R3GW 10296414 Ki = 199.53 nM T79062 D0T2RY 9948320 Ki >= 1000 nM T79062 D0X4PH 11224758 Ki = 0.22 nM T79062 D0X6MT 4106 EC50 = 0.6 nM T79062 D0X7SD 888197 Ki = 156 nM T79062 D0X9YS 23642275 Ki = 0.6 nM T79062 D0XX2U 16006606 Ki = 8.2 nM T79062 D0Y0SA 135399666 EC50 > 10000 nM T79062 D0Y9TL 13702393 Ki = 793 nM T68251 D00HNB 25419 IC50 = 145000 nM T68251 D00MDP 466151 Ki = 0.05 nM T68251 D01UBX 451415 IC50 = 9900 nM T68251 D01XWG 30323 IC50 = 1900 nM T68251 D04AIT 5280445 IC50 = 3610 nM T68251 D07VLY 31703 IC50 = 1100 nM T68251 D0K8KX 5280343 IC50 = 6680 nM T68251 D0Q8CS 60937 IC50 = 7200 nM T68251 D0R9BG 1990 IC50 = 15000000 nM T68251 D0RA5Q 72172 IC50 = 3400 nM T68251 D0S0LZ 54671203 IC50 = 24000 nM T68251 D0V4GY 9552079 IC50 = 7630 nM T68251 D0VM2L 68740 IC50 = 7000 nM T68251 D04LTF 9868980 IC50 = 0.46 ug.mL-1 T68251 D05VZE 119031 IC50 = 0.43 nM T68251 D0F2JS 15547703 IC50 = 190 nM T68251 D0MW3H 9824350 Ki = 154 nM T68251 D0N4IV 10718956 IC50 = 1.7 nM T68251 D0U2BH 65064 IC50 = 9600 nM T68251 D09EFW 46861776 IC50 = 3.42 nM T68251 D0G1LL 74221072 IC50 = 35000 nM T68251 D0LO1Z 5281858 IC50 = 6300 nM T68251 D0N6ZA 74221131 IC50 > 100000 nM T68251 D0UM5R 74221070 IC50 = 4700 nM T68251 D00UCC 9827497 IC50 = 0.78 nM T68251 D01DVX 9847838 IC50 = 482 nM T68251 D03BOZ 3342298 Ki = 0.22 nM T68251 D05VNG 9908389 IC50 = 1.8 nM T68251 D08CEE 10478364 Ki = 200 nM T68251 D0E5GY 9904965 IC50 = 7.4 nM T68251 D0P8YC 5362422 IC50 = 0.73 nM T68251 D0Q1CD 6918336 Ki = 11 nM T68251 D0T2IQ 443600 IC50 = 3000 nM T68251 D0T9HG 132519 IC50 = 0.104 nM T68251 D0Y1XT 128564 Ki < 1 nM T68251 CNA81R 1836 Ki = 80 nM T68251 CQS47H 2299 IC50 = 0.5 nM T68251 CZ45IU 4219 IC50 = 3.6 nM T68251 C24IRS 4222 Ki = 2000 nM T68251 CW1H7U 4323 IC50 = 5.998 nM T68251 CS8X0P 16124 IC50 = 49000 nM T68251 CL2W6Q 38422 IC50 = 7100 nM T68251 CA3M5F 68443 IC50 = 389000 nM T68251 CYEU83 69033 Ki = 70000 nM T68251 C0PY5N 77754 Ki > 100 nM T68251 C5Z1QA 96028 IC50 > 200000 nM T68251 CP4O2C 121255 Ki = 65000 nM T68251 CCY6L8 169853 IC50 = 31400 nM T68251 C7ROG5 177347 IC50 = 91.3 nM T68251 CP7Q8T 240910 Ki = 15000 nM T68251 CX3DK6 283995 Ki = 9000 nM T68251 CBN39D 285263 IC50 = 86.74 nM T68251 COFX01 352863 Ki = 70000 nM T68251 CNM0P3 391527 IC50 = 7 nM T68251 C4U7SY 401129 IC50 = 18700 nM T68251 CV60YH 445010 IC50 = 5 nM T68251 CK9M3P 445018 IC50 = 1 nM T68251 C4D7TS 448002 IC50 = 9.1 nM T68251 CR51PG 448593 Ki = 210 nM T68251 CC54LQ 450256 IC50 > 100000 nM T68251 CG1I8P 467296 IC50 = 88000 nM T68251 CTPW02 467297 IC50 = 34000 nM T68251 C9I8WB 478379 Ki = 0.2 nM T68251 C45JSH 639942 IC50 = 5.28 nM T68251 CP91NX 677915 IC50 = 1649.92 nM T68251 CS4O7K 685005 IC50 > 500000 nM T68251 CDE9V2 689424 IC50 = 1945.82 nM T68251 C5O0TJ 690158 IC50 = 8.95 nM T68251 C7TPR6 690965 IC50 = 5.37 nM T68251 CP1Q6R 703233 IC50 = 61000 nM T68251 C9FL2X 721434 IC50 = 1785.67 nM T68251 CTO15S 727131 IC50 = 9.17 nM T68251 CTV50K 727184 IC50 = 1859.32 nM T68251 C2CL6X 732134 IC50 = 6.32 nM T68251 CPKI76 765318 IC50 = 9.99 nM T68251 CXME85 766168 IC50 = 9.72 nM T68251 CWQG91 770865 IC50 > 1000 nM T68251 CQB03J 780790 IC50 = 6.41 nM T68251 C7EHR1 787183 IC50 = 5.46 nM T68251 C5MF2E 795596 IC50 = 1853.73 nM T68251 C1K0NF 795855 IC50 = 9.13 nM T68251 CW56XG 875024 IC50 = 9.66 nM T68251 C17IXT 910211 IC50 = 9.02 nM T68251 C9IFC6 1348435 IC50 = 2700 nM T68251 C8A5CX 1800786 IC50 = 500 nM T68251 CN9C8D 2140735 IC50 = 350000 nM T68251 C36DGS 2211098 IC50 = 53 nM T68251 CN6E3U 2366268 IC50 = 3600 nM T68251 C1ND5S 2734394 IC50 = 121000 nM T68251 CN62WX 2800809 IC50 > 10000 nM T68251 CEHZ37 3042462 IC50 = 383000 nM T68251 CY3TD6 3348132 Ki = 20 nM T68251 CME24U 3649035 IC50 = 26000 nM T68251 C3EI6T 4085085 IC50 = 67000 nM T68251 CBN96T 4358655 IC50 = 50118.72 nM T68251 CC5O4E 4369384 IC50 = 2000 nM T68251 CP8D7Y 4478236 IC50 = 20 nM T68251 CQ4Y5M 4626827 IC50 = 4.6 nM T68251 CZBY34 5220706 Ki = 72000 nM T68251 C20HRJ 5273475 IC50 = 6.24 nM T68251 CZS0G5 5276565 IC50 > 100000 nM T68251 C3JN0F 5277465 IC50 > 100000 nM T68251 CRJK67 5277481 IC50 = 37400 nM T68251 CYF7S5 5277490 IC50 = 15500 nM T68251 CQ4VL5 5287415 IC50 = 0.8 nM T68251 CW5SE3 5288615 IC50 = 4.7 nM T68251 CJ3QI1 5288814 IC50 = 2905 nM T68251 C5IDT0 5289314 Ki = 115 nM T68251 CVLS16 5319161 IC50 = 3880 nM T68251 CZC3I7 5326979 IC50 = 58000 nM T68251 CL89FO 5496920 Ki = 33 nM T68251 CDI23X 5941957 IC50 > 100000 nM T68251 C1K8FQ 6439677 IC50 = 800 nM T68251 CJG2B7 6476333 IC50 = 8960 nM T68251 CL5DH0 6479915 IC50 = 3580 nM T68251 CQEF36 6539670 IC50 = 1 nM T68251 C1LQD2 6540261 IC50 = 1100 nM T68251 CP7BG0 6852146 IC50 = 5 nM T68251 CN5L2B 6852147 IC50 = 1.5 nM T68251 CP2XK7 6882342 IC50 = 120000 nM T68251 CPFV65 6916013 Ki = 81.28 nM T68251 C7AZE5 6930803 IC50 = 100 nM T68251 C7Y1BX 9543420 IC50 = 13.3 nM T68251 CIJ25V 9794947 IC50 = 20000 nM T68251 CLK61C 9797144 Ki = 73 nM T68251 C7NP9Z 9798247 IC50 = 28 nM T68251 CET56A 9801414 Ki = 10 nM T68251 C76RCQ 9801569 IC50 = 341 nM T68251 C68HMJ 9801786 IC50 = 380 nM T68251 CJY12B 9802219 Ki > 3000 nM T68251 CIXD67 9802768 IC50 = 0.33 nM T68251 CUSD58 9803469 IC50 = 19 nM T68251 C4A0XM 9804305 IC50 = 457 nM T68251 CQ46XD 9804842 IC50 = 8700 nM T68251 CP65QD 9805079 Ki = 482 nM T68251 C1HP7E 9805710 IC50 = 25 nM T68251 CASW18 9806452 Ki = 17 nM T68251 C76CKA 9807105 Ki = 805 nM T68251 CTK6J8 9808181 IC50 = 34200 nM T68251 C9RQM7 9808674 IC50 = 0.3 nM T68251 CTO36D 9817594 IC50 = 30000 nM T68251 C5OE1B 9821883 Ki = 11 nM T68251 CJC20A 9822095 IC50 = 17 nM T68251 C6KJ9W 9822461 IC50 = 8.7 nM T68251 C6IX7G 9822926 IC50 < 0.1 nM T68251 C1MPW9 9823182 IC50 = 19 nM T68251 CTF8V4 9823391 Ki > 3000 nM T68251 CVN5Z3 9823395 IC50 = 12 nM T68251 C1PW5U 9824010 IC50 = 998 nM T68251 CDJB86 9825720 IC50 = 0.1 nM T68251 CXL65P 9825920 Ki > 3300 nM T68251 CL0G8K 9825927 IC50 = 602.56 nM T68251 C65ZHY 9826199 IC50 = 0.61 nM T68251 C1I6KQ 9826286 Ki = 500 nM T68251 C1A7NJ 9827355 Ki = 0.71 nM T68251 C3SZ8Y 9827469 Ki = 1244 nM T68251 C7I2FO 9828039 Ki = 324 nM T68251 C1GR4N 9828276 IC50 > 25000 nM T68251 CC1NG5 9829581 IC50 = 20 nM T68251 C7SRM4 9837496 IC50 = 3000 nM T68251 C9PW7L 9841168 Ki = 28.5 nM T68251 C5XL7R 9841323 IC50 = 0.6 nM T68251 CA7DJ9 9842114 IC50 = 3.199 nM T68251 C32JRZ 9843079 IC50 = 140 nM T68251 C6YT5W 9843479 IC50 = 40 nM T68251 CWY1J9 9846501 Ki > 3000 nM T68251 CE9AL3 9847113 IC50 < 0.1 nM T68251 CA1IP0 9847191 Ki > 3000 nM T68251 C8IMT2 9847787 IC50 = 1.1 nM T68251 C7VXJ5 9848025 IC50 = 3.9 nM T68251 C4IEK0 9850035 IC50 = 0.2 nM T68251 CD1KW6 9851858 Ki = 0.01 nM T68251 C5DGI9 9851911 IC50 = 6.6 nM T68251 C2FYO3 9852206 Ki = 0.01 nM T68251 C5TUJ7 9862317 IC50 = 39 nM T68251 C8GE7U 9862764 IC50 = 59 nM T68251 CS5JT6 9864502 IC50 = 59 nM T68251 CQ0J1G 9865191 IC50 = 17 nM T68251 CI8Z0R 9866250 IC50 = 1.6 nM T68251 CQ9SG1 9866486 IC50 = 1208 nM T68251 CR10NL 9866770 Ki > 3000 nM T68251 C0YN1X 9867935 IC50 = 20 nM T68251 CK3F1T 9868079 IC50 = 1.3 nM T68251 CX57RB 9868249 Ki > 3000 nM T68251 CJS23I 9868333 Ki > 3333 nM T68251 CJ8DP1 9868672 IC50 > 6000 nM T68251 C24JSB 9868858 IC50 = 2 nM T68251 CLQ29X 9869597 IC50 = 262 nM T68251 CG17NZ 9869811 IC50 = 4 nM T68251 CMEA71 9869947 IC50 = 0.5 nM T68251 C38BVX 9870100 IC50 = 19 nM T68251 CZO2I0 9870133 IC50 = 3 nM T68251 CA48SX 9870269 IC50 = 743 nM T68251 CD1XQ2 9871305 IC50 = 1.9 nM T68251 CSM16R 9871355 IC50 = 158 nM T68251 CHU9I8 9871883 IC50 < 1 nM T68251 C5NM6P 9872886 Ki = 91 nM T68251 C0TCJ2 9880675 Ki = 667 nM T68251 CW8IC4 9882151 IC50 > 100000 nM T68251 C0ZT7A 9883002 Ki = 13.9 nM T68251 C75DAZ 9885136 IC50 = 0.65 nM T68251 CG35XZ 9885916 IC50 = 148 nM T68251 CZBK85 9886177 IC50 = 21 nM T68251 C2M4EC 9887473 Ki > 3333 nM T68251 C4PB5Z 9887544 IC50 = 2.6 nM T68251 C3ZG6O 9887870 IC50 = 4 nM T68251 C8AJB7 9888429 Ki > 3000 nM T68251 CVP45O 9888530 IC50 = 175 nM T68251 CDW1O4 9888922 IC50 = 196 nM T68251 CD1U5P 9889190 IC50 = 12 nM T68251 C27HMG 9889517 IC50 = 1.6 nM T68251 C26SZX 9890226 IC50 = 0.4 nM T68251 CWN19T 9890526 IC50 = 3.3 nM T68251 CD79UJ 9890632 IC50 = 92000 nM T68251 CU65HY 9891358 IC50 = 0.06 nM T68251 C3QSE6 9891814 IC50 = 18 nM T68251 CF1X0W 9892321 IC50 = 534 nM T68251 CH69LT 9892815 IC50 < 0.1 nM T68251 CZU7Y4 9892876 IC50 = 73 nM T68251 CK1F3O 9892889 Ki > 305 nM T68251 C1NCU4 9894184 IC50 = 300 nM T68251 CX5G0F 9894469 IC50 = 1300 nM T68251 CZK6O9 9895099 IC50 = 300 nM T68251 CSIB97 9896504 IC50 > 30000 nM T68251 C5DW9S 9902427 IC50 > 30000 nM T68251 C97GSC 9903557 Ki = 1915 nM T68251 CD78ZQ 9907286 IC50 = 0.7 nM T68251 CN6WJ1 9909994 IC50 = 230 nM T68251 CJ3K1I 9910075 IC50 = 1480 nM T68251 CPO8V1 9910282 IC50 = 430 nM T68251 CM2F7R 9910302 IC50 = 1.1 nM T68251 C6NUE9 9910550 IC50 = 0.5 nM T68251 CP4LS8 9910727 IC50 = 87 nM T68251 CT50EC 9912183 Ki = 194 nM T68251 C62VZI 9912382 IC50 = 0.7 nM T68251 C3AZP0 9913479 IC50 = 0.3999 nM T68251 CR98KH 9913488 IC50 = 853 nM T68251 CSZV76 9913881 IC50 = 41 nM T68251 C7ZY1L 9914029 IC50 = 62 nM T68251 CA3FW0 9918908 IC50 = 0.004 nM T68251 CG1A6B 9924640 IC50 > 100000 nM T68251 C4YGT6 9928325 IC50 = 7.5 nM T68251 CK5OV9 9930210 IC50 = 33 nM T68251 C03GVA 9932290 Ki = 210 nM T68251 C1I2FW 9932632 Ki > 3000 nM T68251 CCHZ97 9932731 IC50 = 58000 nM T68251 CDXR37 9933197 IC50 = 0.1 nM T68251 CX17KQ 9933408 IC50 = 29 nM T68251 CF26MY 9934052 Ki > 3000 nM T68251 CA5V8M 9934053 Ki = 433 nM T68251 C57WSD 9934240 IC50 = 7 nM T68251 C65ION 9935032 IC50 = 0.1 nM T68251 CGFD83 9936194 IC50 = 188 nM T68251 C1HRU9 9936228 IC50 = 4.1 nM T68251 C68MQN 9936625 Ki = 435 nM T68251 C9OUC8 9936681 IC50 = 196 nM T68251 CG38KL 9936728 Ki = 1.1 nM T68251 CE59TP 9936926 IC50 = 547 nM T68251 CX7VQ9 9937188 IC50 = 10.96 nM T68251 CLM2R8 9941370 Ki = 3.5 nM T68251 C0IBF2 9941371 Ki = 0.03 nM T68251 CA30JY 9946988 IC50 = 70 nM T68251 CWZC93 9947332 IC50 > 100000 nM T68251 CSN61C 9948296 Ki = 1497 nM T68251 C16HTN 9948666 Ki = 27 nM T68251 CF1DO9 9950475 Ki > 567 nM T68251 CQY54S 9952396 IC50 = 2.1 nM T68251 C8C3DL 9953278 IC50 = 539.51 nM T68251 C16GIN 9953861 Ki > 1267 nM T68251 CR6EX3 9953909 Ki = 446 nM T68251 C8RXN6 9954304 IC50 = 297 nM T68251 C9X0YR 9954867 Ki = 6300 nM T68251 CK9HX0 9955125 IC50 = 0.4 nM T68251 C05HGV 9955795 IC50 = 1.1 nM T68251 C8M2RB 9956613 IC50 > 10000 nM T68251 C3Q2UJ 9956686 IC50 = 0.4 nM T68251 CS73TB 9956692 Ki = 2800 nM T68251 CI5TW9 9956699 IC50 = 529 nM T68251 CN76XI 9957653 IC50 = 1 nM T68251 CVG0O2 9959014 IC50 = 0.9 nM T68251 CN8TK0 9959428 IC50 = 661 nM T68251 CV40RB 9960075 Ki = 391 nM T68251 C9DRB7 9966028 IC50 = 110 nM T68251 C8K5VD 9969928 IC50 > 30000 nM T68251 CFQ15E 9976696 IC50 = 22 nM T68251 C0HL2X 9976697 IC50 = 2.7 nM T68251 C09LSY 9979489 Ki > 3333 nM T68251 CUA65C 9982414 IC50 = 12 nM T68251 CJGR30 9983604 IC50 = 0.5 nM T68251 CILK24 9983687 Ki = 1 nM T68251 CO0TX7 9993891 Ki > 600000 nM T68251 C3KX1B 9998685 Ki = 1 nM T68251 CB2J3S 9999667 IC50 = 10 nM T68251 C8W5UK 9999879 IC50 = 120 nM T68251 C6TO0A 10001582 Ki = 1.5 nM T68251 C59WEK 10001843 IC50 < 0.1 nM T68251 C5HN3L 10001964 IC50 = 222 nM T68251 CP5N4E 10005114 Ki = 43 nM T68251 C6U3CK 10006134 IC50 = 0.5 nM T68251 CA8C6U 10008733 Ki = 0.01 nM T68251 CR7T3J 10009978 Ki = 700 nM T68251 C71YGT 10025307 Ki = 4.7 nM T68251 C6O0MN 10026682 Ki = 5300 nM T68251 C6DGR7 10027203 Ki = 1.5 nM T68251 C4VJX9 10027747 IC50 = 32000 nM T68251 CM52RO 10030422 IC50 = 10 nM T68251 CJR59P 10031295 Ki > 3333 nM T68251 CX2W9O 10037048 IC50 = 200 nM T68251 C7J9ZF 10039403 IC50 = 32 nM T68251 C1X0SA 10041385 Ki = 8 nM T68251 CO39PK 10042482 Ki = 39.81 nM T68251 CW2MK1 10043732 Ki = 46 nM T68251 C7CT4E 10045150 IC50 = 0.34 nM T68251 CHF92V 10047100 Ki = 0.23 nM T68251 CCF5Z4 10047585 IC50 = 0.3 nM T68251 CAN59F 10047708 IC50 = 2.2 nM T68251 CV59KC 10049292 Ki = 340 nM T68251 CLZ87W 10051236 Ki = 1598 nM T68251 CSHD67 10054852 IC50 = 0.4 nM T68251 C42YWK 10055393 IC50 = 229.09 nM T68251 CSW7B3 10067146 Ki = 2.8 nM T68251 C69DPZ 10068042 IC50 = 15800 nM T68251 CD3RL7 10070821 Ki > 10000 nM T68251 CB28NP 10073353 IC50 = 30 nM T68251 CJK0R1 10074190 IC50 = 1 nM T68251 CU7DJ1 10081163 Ki = 77000 nM T68251 C8AEK4 10093420 IC50 = 0.38 nM T68251 C5W4ZA 10094362 IC50 = 300 nM T68251 CA6X2Z 10095338 IC50 = 0.6 nM T68251 CMY3X2 10098158 IC50 = 6.1 nM T68251 C2XV5J 10098250 IC50 = 0.4 nM T68251 C3V2HW 10099112 IC50 = 2 nM T68251 CXV2Y3 10109170 Ki = 433 nM T68251 CY6HZ7 10111132 IC50 = 74900 nM T68251 C0G7IY 10114318 Ki = 1870 nM T68251 C4P1LB 10116618 IC50 = 0.44 nM T68251 CU0D4S 10117481 Ki > 3333 nM T68251 CP5L0W 10117663 Ki > 3300 nM T68251 C7OPQ8 10118047 IC50 = 35 nM T68251 C7A8MI 10120093 IC50 < 0.1 nM T68251 CT4V0P 10120622 IC50 = 0.39 nM T68251 CY2N3D 10127629 Ki > 3330 nM T68251 C1N4MJ 10127670 Ki > 3330 nM T68251 CIL09Z 10127889 Ki > 3330 nM T68251 CYU19P 10127901 Ki > 3330 nM T68251 C07KFI 10128313 Ki > 3330 nM T68251 CB3I6K 10128659 Ki > 3330 nM T68251 C6ZK3A 10128916 Ki > 3330 nM T68251 CH0UW2 10129190 Ki > 3330 nM T68251 CZM7F4 10132758 IC50 = 80000 nM T68251 CDR73P 10135184 Ki > 2128 nM T68251 C7KR3Y 10136680 Ki = 440 nM T68251 CNU93J 10136924 Ki = 450 nM T68251 C1CDF2 10136925 Ki = 340 nM T68251 CJ9EX4 10138303 Ki = 550 nM T68251 CFXC89 10139040 Ki > 3333 nM T68251 CGC6S5 10139402 Ki > 3333 nM T68251 CP8QV4 10140363 Ki = 1920 nM T68251 CU6Y9T 10140438 Ki > 3333 nM T68251 CE75BY 10140776 Ki = 1400 nM T68251 CIH36M 10141214 IC50 = 18 nM T68251 C6MSI0 10141443 IC50 = 33000 nM T68251 CLXF15 10141613 Ki > 3300 nM T68251 C7VF1K 10141614 Ki > 3300 nM T68251 CWB5O4 10142326 Ki > 3300 nM T68251 CL7P6G 10143019 IC50 = 0.098 nM T68251 CPXB21 10143028 Ki > 3333 nM T68251 C23WZR 10143587 Ki > 3300 nM T68251 CZW98O 10156375 Ki = 3.8 nM T68251 CYO8D2 10159633 Ki > 3333 nM T68251 CQ4SJ5 10160197 Ki > 3333 nM T68251 CQ41YI 10161391 Ki > 3333 nM T68251 C7SXD4 10162245 Ki > 3300 nM T68251 CO6PS3 10162900 Ki = 150 nM T68251 CR5H6E 10163627 Ki > 2128 nM T68251 CI9VJ5 10163857 Ki > 3333 nM T68251 CR17PV 10164205 Ki > 3333 nM T68251 CZO5V4 10164317 IC50 < 0.4 nM T68251 CCM0Y8 10165180 Ki = 2167 nM T68251 C5ZO9J 10166232 IC50 = 0.53 nM T68251 C6IW4O 10173876 Ki > 3330 nM T68251 CGB27E 10174981 Ki > 3330 nM T68251 CL47AR 10175070 Ki > 3330 nM T68251 C4ULO6 10175077 Ki > 3330 nM T68251 C4QY3V 10175210 Ki = 3100 nM T68251 C84ZQD 10175219 Ki > 3330 nM T68251 CIT0H4 10175323 Ki > 3330 nM T68251 C95IGP 10175331 Ki = 2170 nM T68251 C4PDJ5 10175366 Ki = 110 nM T68251 CT7U0M 10175426 Ki > 3330 nM T68251 CD4AO0 10180362 IC50 = 2300 nM T68251 CEWF13 10180993 IC50 = 81800 nM T68251 CCX3T6 10183064 Ki > 15000 nM T68251 CDM94B 10183693 Ki > 3300 nM T68251 CHB2D3 10184071 Ki > 3333 nM T68251 C3E9NF 10184537 Ki > 3300 nM T68251 CTDP62 10184579 Ki > 3300 nM T68251 CXQ8N0 10185100 Ki > 3333 nM T68251 CK0P3F 10186536 Ki > 2128 nM T68251 CV7YI1 10186544 Ki > 3300 nM T68251 C51RPY 10195069 Ki > 3330 nM T68251 CCHX74 10195307 Ki = 200 nM T68251 C94KHT 10195527 Ki = 930 nM T68251 CDG35O 10196192 Ki = 370 nM T68251 CY36NO 10196425 Ki > 3330 nM T68251 C1JG5W 10196775 Ki > 3330 nM T68251 CVRZ27 10198038 IC50 = 80 nM T68251 C5CUM9 10202769 Ki > 3333 nM T68251 CX8BS3 10203685 Ki > 3333 nM T68251 CE1LI3 10204303 Ki = 90 nM T68251 C32RAQ 10204620 Ki > 3300 nM T68251 CQFP69 10206106 Ki = 270 nM T68251 CS1CA5 10207780 Ki = 1333 nM T68251 C4K1MJ 10208262 Ki > 2128 nM T68251 CYE02Q 10209301 IC50 = 2.6 nM T68251 CD76KE 10209382 Ki > 3333 nM T68251 CG8FA4 10218128 Ki > 3330 nM T68251 C7Y2US 10218353 Ki > 3330 nM T68251 C1C7AH 10223757 Ki > 3333 nM T68251 CYG10Z 10223774 Ki > 3333 nM T68251 CV5X8A 10224181 IC50 > 30000 nM T68251 CGKU70 10224396 Ki = 240 nM T68251 C7K1OR 10224602 IC50 = 1800 nM T68251 CLH71C 10225319 Ki > 3333 nM T68251 C2X1KF 10226116 Ki = 2566 nM T68251 C9CSG3 10226996 IC50 = 650 nM T68251 CUE63Q 10227853 Ki > 3300 nM T68251 C19DFP 10227854 Ki > 3300 nM T68251 CM7B5T 10228228 Ki > 3333 nM T68251 C7T0WH 10229644 IC50 = 1.1 nM T68251 CD2HP3 10230012 Ki = 1333 nM T68251 CCRM18 10231253 IC50 = 1.2 nM T68251 CCTY95 10237492 Ki > 3330 nM T68251 CQH2U3 10238391 IC50 = 200 nM T68251 CO8M7Q 10239526 Ki > 3330 nM T68251 CCQ9V5 10239716 Ki > 3330 nM T68251 CEO4X5 10239762 Ki > 3330 nM T68251 CU7TQ3 10239803 Ki > 3330 nM T68251 CLAX20 10250594 IC50 = 4.2 nM T68251 C0J3TC 10250722 Ki = 60 nM T68251 CL67DT 10252311 Ki < 2.8 nM T68251 CQJ0R3 10252900 Ki = 0.66 nM T68251 CK9DF5 10253223 IC50 = 12000 nM T68251 CQF3V9 10253673 IC50 = 9 nM T68251 CD8QY2 10253933 IC50 > 10000 nM T68251 CB6SE4 10256227 IC50 = 91 nM T68251 C7HZ1M 10270281 IC50 = 21700 nM T68251 C3XD1E 10271240 IC50 > 100000 nM T68251 C2MES9 10271604 Ki > 100000 nM T68251 CWJ02G 10273315 IC50 > 30000 nM T68251 C0K2ES 10273642 Ki > 3333 nM T68251 CJZP24 10273657 Ki > 3333 nM T68251 CK18DB 10273985 Ki > 2128 nM T68251 CGP97S 10274748 Ki = 140 nM T68251 C13NKU 10275545 Ki > 3333 nM T68251 C1NGV9 10276473 Ki > 3333 nM T68251 CES6A5 10276821 Ki = 1566 nM T68251 C1W7SN 10277073 Ki > 3333 nM T68251 CO18TA 10277120 Ki > 3333 nM T68251 CY6K1G 10277706 Ki > 3300 nM T68251 C2XU3O 10278147 IC50 = 0.67 nM T68251 C3IG0K 10280852 IC50 = 0.2 nM T68251 C80WUO 10282084 IC50 = 0.33 nM T68251 C7TWG0 10289551 Ki > 3330 nM T68251 CJ63ER 10289607 Ki > 3330 nM T68251 CR48SA 10289842 Ki > 3330 nM T68251 CO60CU 10290029 Ki = 2700 nM T68251 CJTV12 10293283 IC50 > 30000 nM T68251 CS69YG 10293394 IC50 = 3500 nM T68251 C89YGA 10295733 Ki > 2128 nM T68251 CDU36Y 10296475 Ki = 520 nM T68251 CTL3Y8 10296608 Ki > 3333 nM T68251 C48IRP 10296785 Ki = 500 nM T68251 CQ1Z0G 10298111 IC50 = 35 nM T68251 CN14MI 10298369 Ki > 3333 nM T68251 CU5E9Z 10299198 Ki = 1357 nM T68251 C25EKM 10299665 Ki > 3300 nM T68251 CQ5BE8 10299709 IC50 = 0.35 nM T68251 C1BR6A 10300063 Ki > 3333 nM T68251 C80VEU 10300077 Ki > 3333 nM T68251 C8U3KW 10301524 IC50 = 0.57 nM T68251 CFAU84 10301584 Ki > 3333 nM T68251 CP5AU1 10302088 Ki > 3333 nM T68251 C63BRA 10303333 IC50 = 34 nM T68251 CE1KM9 10311498 Ki > 3330 nM T68251 CJ15OB 10311501 Ki > 3330 nM T68251 C5F0EV 10311947 Ki > 3330 nM T68251 C4R9ZK 10311997 Ki = 83 nM T68251 CE6MB0 10312141 Ki = 116 nM T68251 C7G6QW 10312268 Ki > 3330 nM T68251 CQ5IT9 10312372 Ki > 3330 nM T68251 CP1GW0 10318094 Ki = 0.57 nM T68251 CIDW49 10319098 Ki > 3333 nM T68251 CF4KT9 10320002 Ki > 3333 nM T68251 CG23FV 10320328 IC50 = 4 nM T68251 CJWH74 10321975 Ki > 3333 nM T68251 CVKT01 10322744 IC50 = 50 nM T68251 CY08WJ 10322755 Ki > 3000 nM T68251 CQH5D4 10324032 IC50 = 0.1 nM T68251 CPI8R0 10324532 Ki = 3 nM T68251 CSFZ76 10325592 Ki = 1376 nM T68251 C1C4VZ 10326004 Ki = 0.9 nM T68251 C7UZA4 10340758 IC50 = 3.2 nM T68251 CCK1A4 10342176 IC50 = 8 nM T68251 CFO74N 10343375 Ki = 430 nM T68251 CJIW74 10343996 IC50 = 0.31 nM T68251 C94ANQ 10347529 IC50 = 0.6 nM T68251 C9FU5G 10362663 IC50 = 1 nM T68251 CWIM61 10364088 IC50 = 756 nM T68251 CL4B2U 10364155 IC50 = 567 nM T68251 CBA5I4 10365560 Ki = 1.1 nM T68251 CH89GT 10365752 IC50 = 3.4 nM T68251 CI0T8K 10366352 Ki > 3333 nM T68251 C6WZ4F 10367355 IC50 = 16 nM T68251 CT81YN 10370089 IC50 = 30 nM T68251 CBTO07 10370226 Ki > 3333 nM T68251 C0IUQ7 10387351 Ki > 3333 nM T68251 CZNT94 10389113 IC50 = 4 nM T68251 CY2G0R 10391428 Ki > 3333 nM T68251 C16BSA 10394828 IC50 = 50 nM T68251 CFKA79 10395015 Ki > 2000 nM T68251 C9HM1A 10402302 IC50 = 76000 nM T68251 CLP05D 10407603 IC50 = 5.2 nM T68251 C98HMP 10413940 Ki = 249 nM T68251 C7K0HG 10414437 Ki = 31 nM T68251 CH1S2G 10414974 Ki = 2.5 nM T68251 C4J7IP 10416507 Ki = 86 nM T68251 C0V9FN 10433382 IC50 = 0.1995 nM T68251 CS32HR 10435935 IC50 = 5.1 nM T68251 C7XE1L 10437629 IC50 = 5000 nM T68251 C5WV1N 10439082 Ki = 1867 nM T68251 C54UDR 10453826 IC50 = 891.25 nM T68251 CQUR30 10454592 Ki = 0.21 nM T68251 C6T8VC 10456675 Ki = 0.6918 nM T68251 C8M9FE 10462640 Ki = 30000 nM T68251 CA7DM9 10474389 IC50 = 0.7 nM T68251 CNQZ36 10483139 Ki = 410 nM T68251 COT6G1 10492779 Ki > 200000 nM T68251 C9KHT4 10495552 Ki = 30 nM T68251 CA7HT2 10498521 Ki = 15 nM T68251 C6KD0A 10498747 IC50 = 1.4 nM T68251 CL8O6I 10500340 Ki = 69 nM T68251 CGK80V 10500816 Ki = 35 nM T68251 CVID65 10500886 Ki = 17.78 nM T68251 CP37WK 10501527 Ki = 17 nM T68251 CK6YN5 10501862 Ki = 6 nM T68251 CZ2UY0 10502046 IC50 = 1 nM T68251 C36OMW 10502172 IC50 = 1 nM T68251 C9QE1B 10502327 Ki = 8 nM T68251 CHOX65 10502351 IC50 = 6.7 nM T68251 C5V8HJ 10502382 IC50 < 0.4 nM T68251 CJZ5T8 10502487 IC50 = 2770 nM T68251 CZ1R5Q 10502869 Ki = 8100 nM T68251 CBNM82 10503128 IC50 < 0.4 nM T68251 CO9S5H 10503708 Ki = 12 nM T68251 C5Y4IA 10504081 IC50 = 104 nM T68251 CD80YF 10504445 IC50 = 0.38 nM T68251 C2C7TE 10504472 IC50 = 2 nM T68251 CT2NM3 10505241 Ki = 19 nM T68251 CK2AB5 10505370 Ki = 2400 nM T68251 CH6S8Y 10505729 IC50 > 10000 nM T68251 C65KOE 10506125 IC50 = 33 nM T68251 C6D7JF 10506147 IC50 = 7 nM T68251 C7S0DB 10506158 IC50 = 16 nM T68251 CNH3L8 10506415 IC50 = 280 nM T68251 CS8V1G 10507004 Ki = 30 nM T68251 CV2T7C 10507137 Ki = 1800 nM T68251 C03MRW 10507152 Ki = 1.2 nM T68251 CDSO53 10507214 IC50 = 8.3 nM T68251 CFJ96A 10507282 Ki = 84 nM T68251 CC6H8T 10507755 Ki = 0.8 nM T68251 C9C5EL 10521197 IC50 = 8.4 nM T68251 CBT12Q 10522080 IC50 = 0.8 nM T68251 CXD8I5 10523292 Ki = 75 nM T68251 CZ36JW 10523383 IC50 = 530 nM T68251 C90HBF 10523728 Ki = 13 nM T68251 CQEH42 10524134 IC50 = 0.7 nM T68251 CYU87N 10524260 IC50 = 0.5 nM T68251 CX6EB7 10524337 Ki = 1800 nM T68251 CQTF46 10524338 Ki = 300 nM T68251 CYB53K 10525912 Ki = 33 nM T68251 CJK6G1 10526509 IC50 < 0.4 nM T68251 CSLO13 10526877 IC50 = 1000 nM T68251 CEK90M 10527263 IC50 = 50 nM T68251 CA83ON 10527749 IC50 = 18 nM T68251 CYGU41 10529315 IC50 = 1475 nM T68251 CBV6X5 10529587 IC50 = 4.4 nM T68251 CGK37L 10529602 Ki = 1.5 nM T68251 CIOJ69 10529720 Ki = 3000 nM T68251 C6PGE1 10530040 Ki = 380 nM T68251 C30UCT 10530499 Ki = 13 nM T68251 CQ82VY 10530944 Ki = 24 nM T68251 CEV6I5 10531005 Ki = 50 nM T68251 CJ2TZ3 10531167 Ki = 19 nM T68251 CS0AD8 10532048 Ki 17 nM T68251 C0WHA9 10546565 Ki = 9 nM T68251 C06NQR 10547080 IC50 = 66 nM T68251 C40ZXE 10547784 Ki = 7 nM T68251 CS10ZB 10549106 Ki = 19 nM T68251 C4PK0U 10549114 IC50 = 2.4 nM T68251 C4TA1K 10549256 IC50 < 0.4 nM T68251 C5JS8L 10549329 Ki = 10 nM T68251 CG27UI 10549756 Ki = 39 nM T68251 C82HQE 10550145 Ki = 6 nM T68251 C7WQ5Z 10550399 IC50 = 1 nM T68251 C1FA6T 10551440 IC50 = 50 nM T68251 CC2FM6 10551489 IC50 = 2391 nM T68251 C5UD0A 10551910 IC50 = 19 nM T68251 C4K3UD 10552661 Ki = 11 nM T68251 CU8QP7 10552732 Ki = 10 nM T68251 COYU34 10553872 Ki = 1900 nM T68251 C0S6GT 10554037 Ki = 16 nM T68251 CSQC42 10554611 Ki = 80 nM T68251 C7P5AW 10554727 Ki = 34 nM T68251 CI8XG0 10554869 IC50 = 8 nM T68251 CYJ41F 10554927 Ki = 3600 nM T68251 CZ41HP 10554978 Ki = 16 nM T68251 CD3R8V 10562830 IC50 = 8.32 nM T68251 CT7O9M 10569678 IC50 = 2 nM T68251 C8RWE4 10569743 IC50 = 36 nM T68251 C0M4VN 10570699 IC50 < 100 nM T68251 CE14GM 10570702 IC50 = 3 nM T68251 CUQ29Z 10571396 Ki = 170 nM T68251 CBXZ79 10572150 IC50 = 6 nM T68251 CPF0R5 10572544 Ki = 20 nM T68251 C21VZS 10573362 IC50 = 1.6 nM T68251 C42IAF 10573603 Ki = 15 nM T68251 CG39CF 10574279 Ki = 13 nM T68251 C8LYR6 10574340 IC50 < 1000 nM T68251 C42BTA 10576058 IC50 < 40 nM T68251 CH7Z2V 10576110 IC50 = 81 nM T68251 CK3JV9 10576740 IC50 = 3.3 nM T68251 CJ7KH8 10578213 Ki = 49 nM T68251 C1KH7E 10578728 IC50 = 9 nM T68251 CK05ZH 10579086 Ki = 0.7 nM T68251 C3R2SO 10580533 Ki = 20 nM T68251 C8J6HS 10591505 Ki = 83.18 nM T68251 CIUO27 10593253 IC50 = 2 nM T68251 CB20LM 10594000 Ki = 18 nM T68251 CUTS47 10594564 IC50 = 33 nM T68251 CN4Y6H 10594565 IC50 = 7 nM T68251 CD65OG 10594830 IC50 = 10.96 nM T68251 CJQY74 10595685 IC50 = 50 nM T68251 CI71CK 10595804 Ki = 10 nM T68251 CYNC76 10596158 IC50 = 12 nM T68251 CD65NF 10597516 Ki = 25 nM T68251 CP2H8O 10597673 Ki = 9 nM T68251 CL7EX4 10598952 IC50 > 1000 nM T68251 CUZ73T 10599048 IC50 = 50 nM T68251 CQCW86 10599579 IC50 < 0.4 nM T68251 CW18QK 10599594 IC50 = 1.2 nM T68251 CR1JI4 10600645 IC50 = 7 nM T68251 CN3E8J 10600844 Ki = 1.3 nM T68251 CJ86TP 10601066 IC50 > 1000 nM T68251 C5WUG1 10601082 Ki = 810 nM T68251 CEJ1U0 10603377 Ki = 18 nM T68251 C5G9MI 10610114 Ki = 120 nM T68251 C84URB 10610500 Ki > 100000 nM T68251 CPW6A4 10617505 IC50 > 1000 nM T68251 CL02BO 10618584 IC50 = 12 nM T68251 C06CAN 10619639 Ki = 12 nM T68251 CV14UH 10619971 Ki = 15 nM T68251 CR69NK 10621302 IC50 = 20 nM T68251 CSQ96T 10621933 Ki = 0.44 nM T68251 CVZ32G 10622447 Ki = 20 nM T68251 CL62YC 10622822 IC50 = 24 nM T68251 CL67UQ 10623250 IC50 = 8 nM T68251 C4FYL1 10623748 IC50 = 34 nM T68251 C6R4EG 10624005 Ki = 2 nM T68251 CR8X1Q 10624346 IC50 = 0.65 nM T68251 CKF6D7 10625329 Ki = 7.3 nM T68251 CGB29T 10625771 IC50 = 0.6 nM T68251 C6H9CT 10626366 Ki = 6900 nM T68251 C70MFZ 10626445 Ki = 18 nM T68251 C5VGB1 10626732 Ki = 21 nM T68251 C3NKC0 10626927 Ki = 17 nM T68251 CA63VQ 10640307 Ki = 36 nM T68251 C7KGM3 10642071 IC50 = 0.3 nM T68251 CI2QB9 10642965 IC50 < 0.4 nM T68251 CM1OZ6 10643325 IC50 = 5.9 nM T68251 C41RKE 10643401 Ki = 10 nM T68251 CUAI71 10643973 Ki = 2 nM T68251 CPYV83 10647658 Ki = 71000 nM T68251 CVX7Q2 10648390 Ki = 11 nM T68251 C4TXZ1 10648776 Ki = 100 nM T68251 C6S1KA 10649216 IC50 > 10000 nM T68251 C07FPQ 10649518 Ki = 55 nM T68251 COT6B8 10650624 Ki = 15 nM T68251 C69SPO 10650906 Ki = 0.6 nM T68251 CT23XW 10650907 Ki = 1.8 nM T68251 C13GKL 10658560 IC50 = 315000 nM T68251 C97KZU 10665624 IC50 = 39 nM T68251 CW1E7L 10667540 IC50 = 310 nM T68251 CF0E6H 10668745 IC50 = 13 nM T68251 CSCL07 10668823 Ki = 6.3 nM T68251 C4HJS1 10669027 Ki = 50 nM T68251 CFYC35 10669215 Ki = 3 nM T68251 C6TC0Z 10669216 Ki = 2.5 nM T68251 C78GYJ 10670529 IC50 = 1.3 nM T68251 C5FWS1 10670820 IC50 = 10 nM T68251 C4QVL0 10670896 Ki = 3 nM T68251 CB1F4G 10671203 IC50 = 110 nM T68251 C3DXN5 10671411 Ki = 0.92 nM T68251 CWB19K 10671441 Ki = 1.4 nM T68251 CXDM24 10671863 Ki = 0.54 nM T68251 C17LYV 10672346 IC50 = 26 nM T68251 CMU74I 10672857 IC50 = 6 nM T68251 CU6Y4O 10674458 Ki = 1600 nM T68251 CXTP56 10688727 IC50 < 1 nM T68251 CU5M1J 10691797 Ki = 42 nM T68251 CSA80H 10692194 IC50 < 1 nM T68251 CS5CL7 10692307 IC50 < 0.4 nM T68251 CR5KF8 10692994 IC50 = 535 nM T68251 CDI12G 10693559 IC50 = 6.8 nM T68251 C8JX1G 10693698 Ki = 3 nM T68251 CVML68 10693881 IC50 = 0.7 nM T68251 CM1T7K 10694510 Ki = 2.6 nM T68251 C7SM1E 10694604 Ki = 3.5 nM T68251 C3E1DX 10695165 IC50 = 4.4 nM T68251 C7ZQM4 10695491 Ki = 0.6 nM T68251 CZGC63 10695865 IC50 = 24 nM T68251 CVQF97 10695971 IC50 = 0.3 nM T68251 CW6CF7 10696226 IC50 = 2 nM T68251 C1YFC3 10696977 IC50 = 9 nM T68251 C4BME8 10697140 IC50 = 23 nM T68251 CBN9K8 10697378 Ki = 22 nM T68251 C1O5CQ 10697393 Ki = 210 nM T68251 CM4AI6 10698165 Ki = 100 nM T68251 C4THQ9 10698311 Ki = 280 nM T68251 C6Y1OU 10698367 Ki = 150 nM T68251 CG5JM9 10698412 Ki = 2.8 nM T68251 C56VSE 10698786 Ki = 1.5 nM T68251 C5E8QF 10707457 Ki = 87 nM T68251 C2GL3A 10714610 Ki = 44 nM T68251 C4IWF2 10714988 IC50 = 6 nM T68251 CO9KV7 10715115 IC50 < 1 nM T68251 C78CKH 10715629 IC50 > 20000 nM T68251 CE1D6G 10716217 IC50 = 3.5 nM T68251 C0ZX6T 10717308 IC50 = 9 nM T68251 C3TGW8 10717400 Ki = 61.66 nM T68251 CZ1M3L 10718058 Ki = 19 nM T68251 CQZ7M8 10718133 Ki = 13 nM T68251 CB96HF 10718916 IC50 > 1000 nM T68251 CN8AK6 10718996 Ki = 0.52 nM T68251 C2IS9D 10719476 Ki = 0.73 nM T68251 CVW81M 10719595 IC50 = 28 nM T68251 CI96XV 10720740 Ki = 14 nM T68251 CIV3P5 10720775 Ki = 760 nM T68251 C65IGZ 10720864 Ki = 21 nM T68251 CTGL64 10721152 Ki = 580 nM T68251 CF46SQ 10721337 Ki = 19 nM T68251 C4J1WN 10721454 IC50 = 0.2 nM T68251 CC1FB8 10721904 Ki = 2.5 nM T68251 CB2QD0 10723468 Ki = 0.9 nM T68251 CO7VP4 10737552 Ki = 18 nM T68251 C51DZG 10737732 IC50 = 11 nM T68251 C1LS5U 10738104 IC50 = 1 nM T68251 CL74TG 10738165 IC50 = 0.4 nM T68251 CB8G2D 10739728 Ki = 15 nM T68251 C4FWC9 10740485 Ki = 66 nM T68251 CKJD45 10741133 IC50 = 450 nM T68251 C0WKL7 10741470 Ki = 10 nM T68251 CPDX27 10741484 IC50 > 1000 nM T68251 C0QT2F 10741956 Ki = 7 nM T68251 CLI7B3 10742101 IC50 > 1000 nM T68251 CKX5R3 10742142 IC50 = 33 nM T68251 C39DPG 10742191 IC50 = 4.8 nM T68251 CHW23E 10742387 IC50 = 20 nM T68251 CY2BZ0 10742536 Ki = 41 nM T68251 C1LF0S 10744337 Ki = 48 nM T68251 CEV8X0 10744751 Ki = 25 nM T68251 CSM9H7 10745124 Ki = 800 nM T68251 C5BZ0J 10745489 Ki = 25 nM T68251 C9ILP3 10745718 IC50 = 31 nM T68251 C4IF2L 10745725 Ki = 25 nM T68251 CK30AE 10745748 Ki = 1.6 nM T68251 CWF50D 10745851 Ki = 21 nM T68251 CE09PI 10757715 IC50 = 6 nM T68251 CA3F1N 10758013 Ki = 43.65 nM T68251 CTKR07 10758266 Ki > 200000 nM T68251 CY9W4M 10760229 IC50 > 1000 nM T68251 CLEG16 10761206 Ki = 30 nM T68251 CDX13Z 10761730 Ki = 13 nM T68251 CA4U7D 10762262 Ki = 18 nM T68251 CP2G0N 10763745 Ki = 0.89 nM T68251 C68THN 10763851 IC50 = 0.3 nM T68251 CM54WS 10764477 Ki = 2400 nM T68251 CAG53Y 10764489 IC50 = 11.4 nM T68251 C7X6EC 10764497 Ki = 1500 nM T68251 CY8LV5 10765345 IC50 = 4.7 nM T68251 C3P2TS 10766036 IC50 = 17 nM T68251 CA6C0Z 10766622 Ki = 0.7943 nM T68251 CN6P1J 10766950 IC50 = 2.2 nM T68251 C0R1ZA 10767025 Ki = 0.64 nM T68251 CWR5Z3 10767105 IC50 = 29 nM T68251 CR4I1E 10767157 IC50 = 6 nM T68251 C7Q2EM 10767236 IC50 = 3 nM T68251 CNT4D0 10767387 Ki = 19 nM T68251 C18QVD 10768090 Ki = 61 nM T68251 C01YKA 10768236 IC50 = 13 nM T68251 CQ7J4I 10769007 IC50 = 12 nM T68251 C6VKJ9 10769394 Ki = 16 nM T68251 CQ6U2Y 10780743 Ki = 19 nM T68251 CIN4A9 10783989 Ki = 20 nM T68251 C15PVT 10785952 Ki = 20 nM T68251 CLAP90 10785969 IC50 = 23 nM T68251 C8AF9L 10787938 Ki = 0.88 nM T68251 C0DFB9 10788617 IC50 = 1 nM T68251 CNAE08 10788733 IC50 = 5 nM T68251 CXQD12 10789326 IC50 = 100 nM T68251 CM74LH 10789594 IC50 = 13 nM T68251 C8EOY6 10790150 Ki = 47 nM T68251 CHWG02 10790787 IC50 = 33 nM T68251 C0NP2Z 10790811 IC50 > 1000 nM T68251 C31EHR 10791372 IC50 = 84 nM T68251 C3P7LZ 10792025 Ki = 1.9 nM T68251 C8D1EN 10792133 IC50 = 3.9 nM T68251 C9VML0 10807861 Ki = 226000 nM T68251 CN8I3Z 10808172 IC50 = 9 nM T68251 CP72JG 10810483 IC50 = 4.8 nM T68251 CT1AI4 10810573 IC50 = 2 nM T68251 CU9F7V 10810684 Ki = 15 nM T68251 CS0O7M 10811110 Ki = 17 nM T68251 C49HCM 10812120 IC50 < 40 nM T68251 CEM1J0 10812918 IC50 < 40 nM T68251 CZB7L2 10812929 IC50 = 1.3 nM T68251 C4TF0K 10813874 IC50 < 0.4 nM T68251 CIUN51 10814028 IC50 = 46 nM T68251 CS7BY4 10816934 IC50 = 4 nM T68251 C3AI5Z 10831752 IC50 = 49 nM T68251 CMX2J7 10832371 IC50 > 1000 nM T68251 CF50HD 10832925 IC50 = 4 nM T68251 COE82D 10833334 Ki = 38.9 nM T68251 C5OG4U 10833497 IC50 = 61 nM T68251 C2A0IX 10833840 IC50 = 46.3 nM T68251 CH90ZB 10834348 IC50 = 14 nM T68251 C9M1JI 10834357 Ki = 10.96 nM T68251 CND0X1 10834889 IC50 = 130 nM T68251 CT3MN0 10837022 Ki = 4.6 nM T68251 CGR16B 10837261 IC50 = 1000 nM T68251 CR0E9Q 10837740 Ki = 3.89 nM T68251 C9H4CP 10838922 Ki = 0.52 nM T68251 CB32OK 10838949 IC50 > 1000 nM T68251 CR50UM 10839419 Ki = 5 nM T68251 CHWQ34 10839761 Ki = 1300 nM T68251 CA76MU 10840059 IC50 = 1160 nM T68251 CPD3L7 10840455 Ki = 32 nM T68251 CR2UX3 10840602 Ki = 94 nM T68251 CL1KG7 10840630 Ki = 24 nM T68251 CI0HR4 10840639 Ki = 39 nM T68251 C6ZSP8 10862104 Ki < 2.8 nM T68251 CQ1L7C 10863755 Ki = 690 nM T68251 C0AQL8 10873958 Ki < 2.8 nM T68251 CBQ70P 10874312 IC50 = 6.3 nM T68251 CLG40T 10874819 IC50 = 260 nM T68251 CXY47P 10875332 IC50 = 383 nM T68251 CJ0LE4 10876254 Ki = 50 nM T68251 CIB8Y1 10884337 Ki = 8 nM T68251 C3AY8O 10885569 IC50 = 20 nM T68251 CAU0I3 10885834 IC50 = 0.9 nM T68251 CDZ04P 10887027 Ki = 11 nM T68251 C7AMS4 10895808 Ki = 49 nM T68251 CPJ0I8 10896934 IC50 = 76 nM T68251 CU7YE0 10896986 IC50 = 0.7 nM T68251 C3FQT7 10903871 Ki = 82 nM T68251 CAF1N8 10906013 IC50 = 2500 nM T68251 CX93MR 10907320 IC50 = 9 nM T68251 CM9G8A 10907701 IC50 = 0.42 nM T68251 C13CJH 10907740 IC50 = 62 nM T68251 C69ZTR 10913644 Ki = 312 nM T68251 C2QR0W 10914151 Ki = 701 nM T68251 C7XE3L 10917417 Ki < 2.8 nM T68251 CGI2T1 10928606 IC50 = 176 nM T68251 CXHA75 10928874 IC50 = 1 nM T68251 CXY4L6 10929354 IC50 = 829 nM T68251 CDSQ41 10929404 IC50 = 106 nM T68251 C1QVT6 10939850 IC50 = 0.93 nM T68251 CWO29J 10940364 IC50 = 13 nM T68251 C89IYC 10948209 Ki < 2.8 nM T68251 CC46WL 10950008 Ki > 3000 nM T68251 C9YOU4 10951375 IC50 = 16 nM T68251 CJI1G0 10951750 IC50 = 1 nM T68251 CNBR78 10952384 IC50 = 8.82 nM T68251 C0A2IR 10958121 Ki = 14 nM T68251 C5HS4F 10961382 Ki = 491 nM T68251 CMY8S6 10961569 IC50 = 1.3 nM T68251 CPA1Q2 10961828 IC50 = 2.8 nM T68251 C30FBA 10970628 Ki = 19 nM T68251 CU2Q8S 10971085 IC50 = 320 nM T68251 CQ68IE 10972732 IC50 = 0.34 nM T68251 CJHO94 10972891 IC50 = 1.7 nM T68251 CTP6I0 10973485 IC50 = 3.6 nM T68251 C9DM0P 10980832 Ki = 11 nM T68251 CL7K8S 10983560 Ki < 3 nM T68251 C3UH2B 10983665 Ki = 647 nM T68251 CR9J5B 10983887 IC50 = 1.7 nM T68251 C68LPK 10983913 IC50 = 1.4 nM T68251 CS7D0Z 10984030 IC50 = 0.72 nM T68251 CV4J2F 10984597 IC50 = 0.3 nM T68251 C0G8TE 10993343 Ki = 11 nM T68251 CW8Z6R 10993677 Ki = 2518 nM T68251 CCX0L6 10994350 IC50 = 3.2 nM T68251 CW0Y6I 10994897 IC50 = 2.4 nM T68251 C3QX0T 11005761 IC50 = 0.45 nM T68251 CJM41O 11006091 IC50 = 1.3 nM T68251 C4PNK3 11006191 IC50 = 1810 nM T68251 C95NXQ 11006894 Ki = 0.64 nM T68251 C7WEZ4 11009332 Ki = 21000 nM T68251 C9WPH7 11016072 Ki = 880 nM T68251 CBE68H 11016073 Ki = 850 nM T68251 CG2DK0 11016448 IC50 < 0.4 nM T68251 C3IYK8 11016511 IC50 = 0.32 nM T68251 CF30UR 11016519 IC50 = 3.78 nM T68251 CODQ51 11016616 IC50 < 0.4 nM T68251 C6IHF5 11026991 IC50 > 8 nM T68251 C3LF1Y 11027584 Ki = 3001 nM T68251 CF5KU1 11027718 IC50 = 1.5 nM T68251 CA49QF 11027968 IC50 = 0.91 nM T68251 CLXZ15 11037377 Ki = 4.3 nM T68251 CT2S0G 11038175 IC50 = 7.4 nM T68251 C3W9IT 11046880 Ki = 408 nM T68251 C5R7JX 11049650 Ki = 1595 nM T68251 CW42KO 11049937 IC50 = 1.9 nM T68251 CQ08SN 11049982 IC50 = 1.8 nM T68251 C23KPN 11050468 IC50 = 2.3 nM T68251 C9RU4I 11059620 IC50 = 2.8 nM T68251 CH8O1E 11060081 Ki = 154 nM T68251 CM6X1E 11061555 Ki > 2000 nM T68251 C1N5PT 11070986 IC50 = 3.2 nM T68251 C18EIZ 11071831 IC50 = 0.6 nM T68251 C43JOG 11080156 Ki = 38 nM T68251 CT3VX4 11080936 Ki = 361 nM T68251 CG0A4C 11081333 IC50 = 25 nM T68251 C05MUK 11081992 IC50 = 1.6 nM T68251 CUNM68 11083152 Ki = 231 nM T68251 CS29GX 11091928 IC50 = 2.8 nM T68251 CE8V9B 11092295 IC50 = 4.22 nM T68251 CR8ZA7 11092551 IC50 = 14 nM T68251 CT2CH7 11092701 IC50 = 9.5 nM T68251 C6R7XB 11092861 Ki = 960 nM T68251 CX69YN 11093502 IC50 = 1.2 nM T68251 CR4V2D 11101785 Ki = 410 nM T68251 C8CK3E 11102531 IC50 = 24 nM T68251 C6G2DI 11111616 Ki = 23 nM T68251 CUK03P 11112062 Ki = 5812 nM T68251 CWV45Z 11112302 Ki < 2.8 nM T68251 CY1SR9 11113744 IC50 = 58.1 nM T68251 CNGP50 11122963 IC50 = 0.35 nM T68251 C8YVE5 11123989 IC50 = 5 nM T68251 CNBG53 11124956 IC50 = 1.6 nM T68251 CX2B6C 11125147 Ki = 450 nM T68251 C9GJ7C 11133809 Ki = 94 nM T68251 C2YBQ7 11134935 IC50 = 7.2 nM T68251 C8DMW5 11135133 IC50 = 83 nM T68251 CD3N8B 11135304 IC50 = 16 nM T68251 CF52TX 11143173 Ki = 1507 nM T68251 CH61QF 11144824 IC50 = 2.4 nM T68251 C8HM2R 11145437 Ki = 75 nM T68251 CHF19X 11146467 Ki = 32 nM T68251 C5WS3E 11147931 IC50 = 1000 nM T68251 CM0QK6 11156328 IC50 = 10 nM T68251 C9H1CW 11156691 IC50 = 16 nM T68251 CD1Q0L 11157488 IC50 = 1590 nM T68251 CZ8KI2 11157757 IC50 = 1500 nM T68251 CM04FR 11168103 IC50 = 10 nM T68251 CVR01T 11168326 IC50 = 7.21 nM T68251 CMKT17 11168614 IC50 = 886 nM T68251 C63CLD 11169065 IC50 = 1200 nM T68251 CD3WL8 11179683 IC50 = 8.4 nM T68251 C2LZ7F 11191803 IC50 = 85 nM T68251 CPA84O 11192618 IC50 = 1630 nM T68251 CCQ6N8 11194666 IC50 = 150 nM T68251 C43ONW 11202395 Ki > 3333 nM T68251 CO76XI 11205873 IC50 = 5000 nM T68251 C9R7OM 11207122 IC50 = 50000 nM T68251 CO87YZ 11215538 IC50 = 5000 nM T68251 CIZW31 11226189 IC50 = 323 nM T68251 C3LEA2 11226622 IC50 = 7 nM T68251 CEL1F0 11248884 IC50 = 19 nM T68251 CUOH67 11252195 IC50 = 500 nM T68251 CJZ3P6 11257884 Ki = 0.4 nM T68251 CO7T3M 11261246 IC50 = 0.41 nM T68251 CWG8Y6 11271094 IC50 = 236 nM T68251 C2OJ8Q 11272747 IC50 = 15000 nM T68251 CJX60I 11284255 IC50 = 5110 nM T68251 C6LJM4 11284404 IC50 = 522 nM T68251 CP17ID 11284983 IC50 = 1700 nM T68251 CF9O2R 11286824 IC50 = 3000 nM T68251 C1IW7N 11292680 IC50 = 0.09 nM T68251 C8C5AV 11294179 Ki > 3333 nM T68251 C7H9JG 11295013 IC50 = 26 nM T68251 C0ZI3J 11298263 IC50 > 200000 nM T68251 C78QSH 11307739 IC50 = 16 nM T68251 CRP08M 11310883 IC50 = 1000 nM T68251 CJ09XO 11317090 IC50 = 5 nM T68251 CK91YW 11317404 IC50 = 68 nM T68251 CLH50U 11318841 IC50 = 1760 nM T68251 C1SN8I 11319030 IC50 = 63 nM T68251 CN2P4G 11328571 IC50 = 321 nM T68251 C9FW7I 11330706 IC50 = 3650 nM T68251 C0XR3B 11330861 IC50 = 3010 nM T68251 CQH57S 11342435 IC50 = 135 nM T68251 CZ8B0D 11349945 Ki < 3.3 nM T68251 CYAK73 11353754 IC50 = 81 nM T68251 CA5P8H 11355488 IC50 = 76000 nM T68251 C7QNX8 11363138 IC50 = 1662 nM T68251 CHG6W0 11365417 IC50 = 62 nM T68251 CM8Y1J 11367571 IC50 = 3000 nM T68251 CTQK48 11373358 Ki > 3333 nM T68251 CLE30X 11374591 IC50 = 2.14 nM T68251 C5KU3Z 11376005 IC50 = 595 nM T68251 CEM0A7 11387990 IC50 = 6200 nM T68251 COZN84 11388372 IC50 = 15 nM T68251 CUJ4V0 11391937 IC50 = 8.2 nM T68251 C9ABX8 11397130 Ki > 3333 nM T68251 CF78WB 11398934 IC50 = 1410 nM T68251 C13NCF 11400989 IC50 = 300 nM T68251 CZM5E8 11410471 IC50 = 30 nM T68251 CU04HF 11419551 IC50 = 47 nM T68251 C4K9DO 11421151 IC50 = 3.2 nM T68251 C30PFC 11421763 IC50 = 2060 nM T68251 CK95HW 11429232 Ki = 0.4 nM T68251 C01FLQ 11441438 Ki = 3.2 nM T68251 CFE6A0 11443957 IC50 = 37 nM T68251 CZY3W9 11444262 IC50 = 12 nM T68251 CI0V6L 11447356 IC50 = 4000 nM T68251 COS67B 11456566 IC50 = 1370 nM T68251 CCMT46 11457732 IC50 = 20 nM T68251 C96DRO 11466734 IC50 = 581 nM T68251 C7QF0G 11467517 IC50 = 2150 nM T68251 CQ1D6E 11470070 IC50 = 200 nM T68251 C1KP2Q 11473879 Ki > 3333 nM T68251 CZBF91 11476645 IC50 = 156 nM T68251 C5Z4UP 11504653 IC50 > 2000 nM T68251 CWS35C 11510523 IC50 = 1270 nM T68251 C5G8PM 11511807 IC50 > 2000 nM T68251 C5VUM2 11517085 Ki = 300 nM T68251 C43OXZ 11519233 IC50 = 9 nM T68251 C5MO0U 11526826 IC50 = 5.3 nM T68251 CI8R5J 11529867 IC50 = 23100 nM T68251 C9Y6LH 11533683 IC50 = 3270 nM T68251 CE01PG 11543178 IC50 = 15370 nM T68251 C2OA3K 11547967 IC50 = 546 nM T68251 C1NZB9 11548265 IC50 = 0.3 nM T68251 CIWP38 11555036 IC50 = 18 nM T68251 C47VIT 11562805 IC50 = 4000 nM T68251 C61BQP 11562817 IC50 = 1563 nM T68251 CO9BC3 11562986 IC50 = 1272 nM T68251 CW5A4S 11569716 IC50 = 6.3 nM T68251 CHV2G1 11575995 Ki > 10000000 nM T68251 C3H2DG 11577137 IC50 = 135 nM T68251 CM6GO2 11577517 IC50 > 2000 nM T68251 CXT05D 11581283 IC50 = 1120 nM T68251 CX2PQ5 11588332 IC50 = 5740 nM T68251 C0Q5FU 11592023 IC50 > 2000 nM T68251 CSQ5M8 11598899 IC50 = 264 nM T68251 CTQ87G 11599024 IC50 = 1440 nM T68251 COT65V 11599397 IC50 > 2000 nM T68251 CUL5H2 11605631 IC50 = 4 nM T68251 CQ7G5D 11613116 IC50 = 1999 nM T68251 C0VCJ8 11613810 IC50 = 3.6 nM T68251 CXKU59 11620780 IC50 > 5000 nM T68251 CCBS59 11634234 IC50 = 280 nM T68251 CZO71U 11639846 IC50 = 550 nM T68251 CNY92D 11640694 Ki > 30000 nM T68251 CFV49P 11641262 IC50 < 1.5 nM T68251 CH3V8F 11663480 IC50 > 2000 nM T68251 CR2UN0 11669859 IC50 = 7.4 nM T68251 CK9F4P 11673778 IC50 = 9000 nM T68251 C90GCV 11675055 IC50 = 2110 nM T68251 C0WV8R 11678029 IC50 > 2000 nM T68251 CFC74O 11678245 IC50 = 574 nM T68251 C28WNK 11682752 Ki = 16 nM T68251 CY0T4D 11685065 IC50 > 2000 nM T68251 CRF7V9 11691964 IC50 = 1.3 nM T68251 CKGR97 11692294 IC50 = 1999 nM T68251 C6ORK5 11692747 IC50 = 655 nM T68251 C3U6ZR 11697504 Ki = 33000 nM T68251 C4BGI2 11698938 IC50 = 6958 nM T68251 C6PM1J 11713686 IC50 = 1380 nM T68251 C1MJ3P 11713694 IC50 = 126 nM T68251 C2BJ3X 11716217 Ki = 4599 nM T68251 C4FU2H 11717997 IC50 = 3430 nM T68251 C4ECU2 11720597 IC50 = 315 nM T68251 CCD93H 11730086 Ki = 80 nM T68251 C68KBY 11732585 Ki = 85 nM T68251 C7CED0 11733417 IC50 = 549 nM T68251 CI0KL2 11733573 IC50 = 13 nM T68251 C64LQC 11733862 Ki > 3000 nM T68251 CIU03K 11734219 Ki = 332 nM T68251 CJOE40 11748355 Ki = 4.8 nM T68251 C4HD9K 11751106 IC50 = 271 nM T68251 CG8U3H 11753351 IC50 = 3810 nM T68251 CO8QT0 11753905 Ki = 1100 nM T68251 C3P0TZ 11754739 Ki = 238 nM T68251 CJ4G5D 11754907 IC50 = 16.2 nM T68251 CD6S0B 11757331 IC50 > 100000 nM T68251 C5E7KU 11757592 Ki = 0.6 nM T68251 CUC9R5 11758082 IC50 = 0.7 nM T68251 CF2J8V 11758099 IC50 = 1000 nM T68251 CQ3Y4E 11761293 IC50 = 110 nM T68251 C6K8HR 11761578 Ki = 136 nM T68251 C04DFH 11783486 Ki = 4.8 nM T68251 CQP12F 11787159 IC50 = 86 nM T68251 C7BV5P 11792968 Ki = 40.74 nM T68251 CV16JZ 11793588 IC50 > 1000 nM T68251 CCSD72 11795621 IC50 = 7.8 nM T68251 CY8N1U 11795715 Ki = 5 nM T68251 CY7H2T 11795824 Ki = 12 nM T68251 C3DE6J 11796352 IC50 = 5.4 nM T68251 CK24XT 11796481 Ki = 8 nM T68251 C46KHU 11796490 IC50 = 5.2 nM T68251 C47OIA 11797154 IC50 = 0.8 nM T68251 CJ4VL3 11797382 IC50 = 10 nM T68251 C7VLP9 11798303 IC50 < 200 nM T68251 CHQR96 11798386 IC50 < 0.4 nM T68251 CZ3C9P 11798873 IC50 = 1.5 nM T68251 CXFP23 11798966 IC50 = 3.311 nM T68251 C19RCP 11799753 Ki = 3.7 nM T68251 CHS4I2 11800528 Ki = 38 nM T68251 CZ5LP1 11800650 IC50 = 10 nM T68251 CQ9HE2 11811551 IC50 = 53 nM T68251 CK03NI 11811717 Ki = 35 nM T68251 CLW3F1 11812791 IC50 = 24.2 nM T68251 C20PYA 11813392 IC50 = 12 nM T68251 CH3SV6 11813493 IC50 = 76 nM T68251 C8DY3Z 11817193 IC50 = 1000 nM T68251 CEN02U 11822212 Ki = 75 nM T68251 CDU9S2 11824087 Ki = 52 nM T68251 C3VO5H 11824148 Ki = 0.3 nM T68251 CKEM29 11827006 IC50 = 46 nM T68251 CV2MX4 11832221 Ki = 108 nM T68251 C48QEH 11833533 Ki < 2.8 nM T68251 CI2OP1 11942810 IC50 = 2700 nM T68251 C4XR5G 11963536 IC50 = 664 nM T68251 C02BWA 11967143 Ki > 2000 nM T68251 CB80OT 12000718 IC50 > 20000 nM T68251 C43PJZ 12000720 IC50 > 20000 nM T68251 CN72PQ 12037467 IC50 = 82.17 nM T68251 CKI97Z 12344252 IC50 > 200000 nM T68251 C0K8ZX 12404978 IC50 > 500000 nM T68251 C0JID3 12447203 Ki > 100000 nM T68251 CKSL53 12507616 IC50 > 200000 nM T68251 CTHQ39 12635073 Ki = 14000 nM T68251 CIQX87 12635074 Ki = 72000 nM T68251 C0XKJ1 12671872 IC50 = 1000 nM T68251 COF8W3 13008156 IC50 > 200000 nM T68251 CC9DK6 13384604 IC50 = 300 nM T68251 CSR94V 13559594 IC50 = 3.28 nM T68251 C71ASU 13644537 IC50 = 8.22 nM T68251 CQTX49 13738810 IC50 > 100000 nM T68251 CVH7N1 13746652 IC50 = 9800 nM T68251 C1AJO7 13968141 IC50 > 300000 nM T68251 CP8L5J 14104451 IC50 = 2000 nM T68251 CLS53V 14151811 IC50 = 9500 nM T68251 CQ3D9C 14151815 IC50 = 18000 nM T68251 C8TH1O 14177156 IC50 > 500000 nM T68251 CM9PD5 14237653 IC50 = 12400 nM T68251 CA2H8V 14303060 IC50 = 170 nM T68251 C7KDL3 14616290 IC50 = 98020 nM T68251 CY4XO2 14616291 IC50 > 500000 nM T68251 C1Q5JU 14616298 IC50 = 67010 nM T68251 C9TF7I 14616299 IC50 = 246260 nM T68251 CHU6J5 14616300 IC50 = 81010 nM T68251 C86DNV 14616301 IC50 = 64300 nM T68251 C47DQP 14732854 IC50 = 19000 nM T68251 C1IZ7D 15296597 Ki = 15 nM T68251 CGH19T 15296844 IC50 > 300000 nM T68251 CSU04W 15406874 IC50 = 5.8 nM T68251 C63MFQ 15435266 IC50 = 3 nM T68251 CH80JI 15435267 Ki = 25 nM T68251 CZ0NL1 15484680 IC50 = 6 nM T68251 CT68FI 15487434 Ki = 120 nM T68251 CJR3Z8 15487435 Ki = 110 nM T68251 C46XNB 15487436 Ki = 560 nM T68251 CP2C4Z 15524387 Ki = 31600 nM T68251 CAF7R5 15524388 Ki = 52 nM T68251 C17HGN 15524389 Ki = 6600 nM T68251 CFH8Y6 15524390 Ki = 35000 nM T68251 C3N1KV 15629940 IC50 > 100000 nM T68251 CVUY27 15631189 IC50 = 8490 nM T68251 C5TLB4 15765753 IC50 = 3.97 nM T68251 C5FA3L 15871222 IC50 = 0.7 nM T68251 CB3A4Z 15941413 Ki = 78 nM T68251 CA40FE 15941550 Ki = 6 nM T68251 CM3D1L 15941553 Ki = 110 nM T68251 CQ0ZL7 15941677 Ki = 23 nM T68251 C6F9WV 15941679 Ki = 70 nM T68251 C7C1HI 15941680 Ki = 34 nM T68251 CU2C1R 15987326 IC50 = 1040 nM T68251 CL7KX3 16040152 IC50 = 3 ug.mL-1 T68251 CTZ3R1 16040153 IC50 = 12.4 ug.mL-1 T68251 C4VW5F 16058482 IC50 = 35 nM T68251 C4WX2I 16108938 IC50 > 1000 nM T68251 CD51GI 16108939 IC50 = 5 nM T68251 C5YVB0 16108940 IC50 = 446 nM T68251 CB4DU9 16108941 IC50 > 5000 nM T68251 CBW71J 16108942 IC50 > 5000 nM T68251 CG6R9L 16108943 IC50 = 960 nM T68251 CN62KM 16108944 IC50 = 150 nM T68251 C7YS5Q 16108947 IC50 = 200 nM T68251 CLD2Y4 16108948 IC50 > 5000 nM T68251 CJR95O 16108949 IC50 > 1000 nM T68251 CRQ26L 16108950 IC50 = 350 nM T68251 CH80AG 16108951 IC50 = 13 nM T68251 CWB0G9 16108952 IC50 = 64 nM T68251 CS46XU 16126723 IC50 = 1.2 nM T68251 CC6OH2 16129741 IC50 = 43200 nM T68251 CH7D2Q 16420684 IC50 = 21200 nM T68251 C91EXN 16655061 IC50 = 555 nM T68251 CQS0F5 16719301 IC50 = 180 nM T68251 C0OUC6 16726064 IC50 = 23000 nM T68251 C75XDI 16730519 IC50 > 2000 nM T68251 C2W1VA 16739287 Ki = 5000 nM T68251 C6F9LM 16748789 IC50 > 30000 nM T68251 CXB10H 16748901 IC50 > 100000 nM T68251 C7YJZ5 17748252 IC50 = 2200 nM T68251 C3S2TQ 17754305 IC50 = 431 nM T68251 CQG89Z 17853548 IC50 = 64190 nM T68251 C2ZAX1 18002715 Ki > 3300 nM T68251 C12UGK 18002722 Ki > 3300 nM T68251 C0IYW8 18002726 Ki > 3300 nM T68251 C8N1DM 18002729 Ki > 3300 nM T68251 CCG96A 18002736 Ki > 3300 nM T68251 C5MLG1 18002745 Ki > 3300 nM T68251 CXT4H2 18002752 Ki > 3300 nM T68251 C26WHK 18002758 Ki > 3300 nM T68251 CV90XS 18002764 Ki > 3300 nM T68251 C8KPM7 18002765 Ki > 3300 nM T68251 CMJ0K3 18002771 Ki > 3300 nM T68251 C2CO9Z 18002775 Ki > 3300 nM T68251 CK8FS7 18173159 IC50 = 6 nM T68251 CX10BM 18173179 IC50 = 24 nM T68251 CQO70Y 18173222 IC50 = 82 nM T68251 C6F8WH 18319167 IC50 = 6 nM T68251 C57FQG 18319202 IC50 = 1790 nM T68251 CJ8G9A 18319234 IC50 = 334.97 nM T68251 CE4J1B 18319263 IC50 = 1300 nM T68251 CXG1K2 18363133 IC50 > 10000 nM T68251 C37BNA 18363136 IC50 > 10000 nM T68251 C0KOW7 18363142 IC50 > 10000 nM T68251 CP04KS 18363146 IC50 > 10000 nM T68251 CLZD96 18363152 IC50 > 10000 nM T68251 CW3KB9 18363153 IC50 > 10000 nM T68251 CK30ZO 18363159 IC50 > 10000 nM T68251 CZU27R 18363164 IC50 > 10000 nM T68251 CC0UV8 18363169 IC50 > 10000 nM T68251 CR3CQ4 18363187 IC50 > 10000 nM T68251 CH5IU9 18363209 IC50 > 10000 nM T68251 CJGZ27 18363210 IC50 > 10000 nM T68251 CWI2A9 18363212 IC50 > 10000 nM T68251 C31LQZ 18363213 IC50 > 10000 nM T68251 CE60WD 18363216 IC50 > 10000 nM T68251 C3L6DU 18363223 IC50 > 10000 nM T68251 CI53DY 18379040 Ki > 3333 nM T68251 CB1U5T 18379077 Ki > 3333 nM T68251 CSX97G 18379115 Ki > 3333 nM T68251 CJHL25 18379123 Ki > 3333 nM T68251 CR0B8G 18379149 Ki > 3333 nM T68251 CS4V5K 18379187 Ki > 3333 nM T68251 CCTY94 18379210 Ki > 3333 nM T68251 CA6K5S 18379235 Ki > 3333 nM T68251 CCSK49 18379254 Ki > 3333 nM T68251 CP4T7S 18379435 Ki > 3333 nM T68251 C9Y5GX 18379443 Ki > 3333 nM T68251 CXL6T9 18379569 IC50 = 173 nM T68251 CKY98M 18379668 IC50 = 9 nM T68251 CSY0N8 18394511 IC50 > 300000 nM T68251 C9J8IN 18445902 IC50 = 800 nM T68251 C5B9WG 18533077 IC50 = 800 nM T68251 C50AEZ 18616892 IC50 = 23.5 nM T68251 CYA3H7 18790040 IC50 > 10000 nM T68251 CBN28Y 18790155 Ki = 270 nM T68251 C03CET 18914685 Ki = 2000 nM T68251 CIEH93 19382975 IC50 = 6400 nM T68251 C60WKH 20196702 IC50 = 5.09 nM T68251 CK8MP3 20620240 Ki = 230 nM T68251 CPC4G6 20620273 Ki = 410 nM T68251 C26UJT 20620561 IC50 = 16 nM T68251 C2E3CY 20620614 IC50 = 48 nM T68251 CVEX54 20620688 IC50 = 6.6 nM T68251 CV1SD8 20620714 IC50 = 11 nM T68251 C3GAC4 20620715 IC50 = 270 nM T68251 C7QV8K 20620757 IC50 = 1100 nM T68251 CVO73Y 20620827 IC50 = 450 nM T68251 CQ14NY 20620831 IC50 = 940 nM T68251 C5RQ8A 20620860 IC50 = 10 nM T68251 CPK09X 20651316 IC50 = 1.4 nM T68251 CG1BD4 20689551 IC50 = 180 nM T68251 C48TWB 20728102 IC50 > 2000 nM T68251 C18RXS 20735191 IC50 < 0.1 nM T68251 C4I1OM 20735209 IC50 = 400 nM T68251 CF1CK9 20735364 IC50 = 0.5 nM T68251 CW3D7O 20760308 Ki = 1002 nM T68251 C09JTR 21130554 IC50 = 0.2 nM T68251 C6VP1T 21130556 IC50 = 0.2 nM T68251 C15UGO 21130558 IC50 = 5 nM T68251 C9H3IG 21130559 IC50 = 1.3 nM T68251 C8Q2OD 21130561 IC50 = 1.3 nM T68251 C25FAD 21130562 IC50 = 0.2 nM T68251 CW2Q5A 21130590 IC50 = 79.98 nM T68251 C9HMC0 21130591 IC50 = 184 nM T68251 CT87YK 21699971 IC50 = 5200 nM T68251 CH4G5T 21699977 IC50 = 400 nM T68251 CQ1GI3 21699983 IC50 = 650000 nM T68251 CJZ58F 21699985 IC50 = 37000 nM T68251 CA3WG1 21699989 IC50 = 4 nM T68251 CE72FU 21700004 IC50 = 950000 nM T68251 CRG8J9 21700008 IC50 = 20 nM T68251 C5JC6W 21700038 IC50 = 160000 nM T68251 CY18IE 21700054 IC50 = 89 nM T68251 CW1YS9 21700072 IC50 = 20 nM T68251 C3QAP8 21700080 IC50 = 45000 nM T68251 CG0RI5 21700124 IC50 = 5900 nM T68251 CR81NU 21700137 IC50 = 1300 nM T68251 CJ4C3K 21700144 IC50 = 85 nM T68251 C94FZS 21700146 IC50 = 26 nM T68251 CXME27 21700151 IC50 = 3400 nM T68251 CFK4Y7 21700160 IC50 = 6900 nM T68251 CIJ93L 21700163 IC50 = 25000 nM T68251 CN80JR 21700178 IC50 = 4 nM T68251 CB1QH3 21700191 IC50 = 480000 nM T68251 CUVE24 21700204 IC50 = 260000 nM T68251 CM42ZR 21700258 IC50 = 4 nM T68251 CMW12T 21700264 IC50 = 1 nM T68251 CKAJ52 21867770 IC50 = 0.7 nM T68251 C45UGA 21996090 IC50 = 16 nM T68251 CIC4S9 22004232 IC50 = 3.4 nM T68251 C36WFA 22096205 IC50 > 100000 nM T68251 CO91AD 22341241 Ki > 3333 nM T68251 CE5DH1 22484408 IC50 = 1.8 nM T68251 CZT05X 22484417 Ki = 550 nM T68251 CZT64B 22484431 Ki = 410 nM T68251 C1O7RC 22485248 IC50 = 400 nM T68251 CAM10T 22485252 IC50 = 0.8 nM T68251 CBJS34 22485260 IC50 < 0.1 nM T68251 C9MU7N 22485263 IC50 = 4.4 nM T68251 CEGJ03 22485276 IC50 = 3.3 nM T68251 C7VB8G 22485289 IC50 = 0.5 nM T68251 CNB02I 22485291 IC50 < 0.1 nM T68251 CAY3N6 22485292 IC50 = 1 nM T68251 C94OCJ 22485302 IC50 = 0.1 nM T68251 C3YL5X 22485311 IC50 = 0.1 nM T68251 C80RSQ 22485314 IC50 = 0.1 nM T68251 CWA03L 22485327 IC50 = 0.2 nM T68251 C6JRW5 22485340 IC50 = 0.1 nM T68251 C5JZF1 22485344 IC50 = 0.35 nM T68251 CI7MY5 22485346 IC50 = 0.1 nM T68251 CI1YL7 22485347 IC50 = 0.25 nM T68251 C25OBD 22485356 IC50 = 0.3 nM T68251 C7I0EW 22485367 IC50 = 0.2 nM T68251 CL64TJ 22485368 IC50 = 0.2 nM T68251 CT4GF9 22485381 IC50 = 6350 nM T68251 C27NDB 22485386 IC50 = 1.7 nM T68251 CTJ9I3 22485392 IC50 = 0.3 nM T68251 C3MG9P 22485396 IC50 = 0.4 nM T68251 CZY10U 22485408 IC50 = 0.3 nM T68251 C89AGT 22485413 IC50 = 0.2 nM T68251 C03NLM 22485417 IC50 = 0.1 nM T68251 C8GHU9 22485432 IC50 = 0.2 nM T68251 C9BT5F 22626996 IC50 = 77 nM T68251 C2Q4XK 22707806 IC50 = 0.1 nM T68251 CD4Z6P 22707833 IC50 = 3500 nM T68251 CMYK90 22707860 IC50 < 0.1 nM T68251 CVF9M4 22922043 IC50 = 23320 nM T68251 CX2JO7 22950015 IC50 = 335 nM T68251 COCN69 22956916 Ki = 1111 nM T68251 C85PXN 22956934 Ki = 771 nM T68251 CIYA45 22985930 IC50 < 0.1 nM T68251 CF75MS 23017979 IC50 = 60000 nM T68251 CQJ3S4 23018008 IC50 = 30000 nM T68251 CM5H2P 23061661 IC50 > 10000 nM T68251 C97LAR 23061665 IC50 > 10000 nM T68251 C2DG6O 23288322 Ki = 2000 nM T68251 C5XW9M 23310222 IC50 = 9 ug.mL-1 T68251 C9IW3E 23433373 IC50 = 1000 nM T68251 CX32YK 23513795 IC50 = 19 nM T68251 C6IZ1S 23513821 IC50 = 113 nM T68251 CPNM93 23513825 IC50 = 62 nM T68251 CML90Q 23513831 IC50 = 54 nM T68251 C87RTM 23513845 IC50 = 249 nM T68251 C4R2AJ 23625454 IC50 = 513 nM T68251 CD3U8A 23627203 Ki = 1300 nM T68251 C8UIC6 23644662 Ki > 100000 nM T68251 CCLA40 23644663 Ki > 100000 nM T68251 CSZ6J4 23645528 Ki = 3.2 nM T68251 C6UH9Q 23645529 Ki = 0.8913 nM T68251 CD0JP3 23645530 Ki = 0.7943 nM T68251 CM37EC 23645531 Ki = 2.399 nM T68251 C9PD5F 23645532 Ki = 2.884 nM T68251 C1OE7R 23645533 Ki = 0.7943 nM T68251 CCSN04 23645534 Ki = 1.4 nM T68251 CU08WI 23645535 Ki = 0.6918 nM T68251 CY41UC 23645536 Ki = 15 nM T68251 CX15EH 23645537 Ki = 3.7 nM T68251 CD3Q6G 23645538 Ki = 12 nM T68251 CE6NQ2 23645539 Ki = 19000 nM T68251 C4VK3U 23645540 Ki = 14000 nM T68251 C8VM1C 23645541 Ki = 73000 nM T68251 C0MUT6 23645542 Ki = 21000 nM T68251 CNI07H 23645543 Ki = 23000 nM T68251 CHK2X1 23645544 Ki = 38000 nM T68251 CW1V2Z 23645545 Ki = 14000 nM T68251 C6SP7T 23645546 Ki = 11000 nM T68251 CD9QO2 23645547 Ki = 900 nM T68251 C25YLZ 23645548 Ki = 90 nM T68251 CL1KC0 23652834 IC50 = 8.37 nM T68251 CL24JR 23655078 IC50 = 940 nM T68251 COIZ43 23655713 IC50 = 4350 nM T68251 CURM98 23655714 IC50 > 100000 nM T68251 CO90JC 23655717 IC50 = 5590 nM T68251 C3M2NQ 23655718 IC50 = 207 nM T68251 C56NMQ 23655910 IC50 = 9110 nM T68251 C9QZX5 23655911 IC50 = 6120 nM T68251 CA8W3K 23656106 IC50 = 239 nM T68251 CU4R7T 23656291 IC50 = 4 nM T68251 CVZ2M1 23656293 IC50 = 22 nM T68251 CL5C1I 23656295 IC50 = 30 nM T68251 CZP12E 23656450 IC50 = 2 nM T68251 CA2PY5 23657418 IC50 = 335 nM T68251 CN9TY1 23657419 IC50 = 992 nM T68251 C9FHZ1 23657421 IC50 = 19 nM T68251 CY9LF1 23657422 IC50 = 8 nM T68251 C28SPW 23657691 IC50 = 41000 nM T68251 CVJ1T7 23657695 IC50 = 20000 nM T68251 CAL05Q 23657697 IC50 = 35000 nM T68251 C6AW7U 23692637 IC50 = 2000 nM T68251 C7KF1N 23729138 IC50 = 6.8 nM T68251 C35QME 24742028 IC50 = 3 nM T68251 CY6KA0 24755074 IC50 = 5000 nM T68251 CG3J2L 24768528 IC50 = 120 nM T68251 CQCJ17 24768595 IC50 = 0.53 nM T68251 C5M3YW 24799779 Ki = 1000000 nM T68251 CWLT01 24806172 IC50 = 61 nM T68251 CN59KZ 24806173 IC50 = 1233 nM T68251 CH4X8K 24806175 IC50 = 13 nM T68251 C9RW0A 24806176 IC50 = 5.2 nM T68251 C18FRG 24807817 IC50 > 100000 nM T68251 CW3X0F 24852010 IC50 = 5.6 nM T68251 C2U0NS 24852011 IC50 = 8.3 nM T68251 C6YPS8 24852048 IC50 = 5 nM T68251 CUK6F1 24852487 IC50 = 95.9 nM T68251 C0MPV5 24852489 IC50 = 59.4 nM T68251 CK0CI6 24860421 IC50 = 334 nM T68251 CZI59C 24860423 IC50 = 97 nM T68251 CE29HI 24860424 IC50 = 1530 nM T68251 CT10JE 24860425 IC50 = 216 nM T68251 CRC98J 24860426 IC50 = 46 nM T68251 C8MKR0 24860427 IC50 = 1312 nM T68251 C3S6DX 24860428 IC50 = 56 nM T68251 C2LNE4 24860429 IC50 = 4181 nM T68251 CF4D0X 24860430 IC50 > 1666 nM T68251 CNR3U7 24866945 IC50 > 100000 nM T68251 CRZ7Y6 24868315 IC50 = 1.8 nM T68251 CFL04M 24881245 IC50 > 300000 nM T68251 CLIC14 24881246 IC50 = 60000 nM T68251 C3U8ZQ 24882385 IC50 = 230 nM T68251 C02WIB 24882535 IC50 = 20 nM T68251 C4FI5C 24901479 IC50 = 40 nM T68251 C6F0ZP 24901485 IC50 = 4.6 nM T68251 C4SP3O 24936157 IC50 = 0.67 nM T68251 CBUA83 24936183 IC50 = 12.6 nM T68251 CQ2K9H 24936215 IC50 = 488 nM T68251 C0EA5F 24936382 IC50 = 0.04 nM T68251 C78OAU 24944977 IC50 = 114 nM T68251 CO6CJ5 24945161 IC50 = 3600 nM T68251 C1C0NX 24945244 IC50 = 5300 nM T68251 CLTQ28 24945246 IC50 = 250 nM T68251 C7ZA6S 24945247 IC50 = 380 nM T68251 CH3O0V 24951588 IC50 = 83 nM T68251 C8I4PT 24951589 IC50 = 17 nM T68251 C2Q1BK 24951590 IC50 = 11 nM T68251 COMJ45 24951950 IC50 = 333 nM T68251 C3JGU2 24951952 IC50 = 24 nM T68251 CC7U2T 24951953 IC50 = 12 nM T68251 CV86KA 24952316 IC50 = 27 nM T68251 CYJ2E9 24952318 IC50 = 2535 nM T68251 CYKM71 24952674 IC50 = 139 nM T68251 C7MC8J 24952678 IC50 = 9.2 nM T68251 C0ZB8O 24953024 IC50 = 5.7 nM T68251 C5Z8XR 24953380 IC50 = 47 nM T68251 C2LN5E 24953381 IC50 = 119 nM T68251 CT2N3H 24953730 IC50 = 9.9 nM T68251 C1KH2Q 24953731 IC50 = 8.6 nM T68251 C0Q5BT 24954067 IC50 = 5.5 nM T68251 C6FI8O 24954068 IC50 = 5.6 nM T68251 CN29BR 24954070 IC50 = 5.5 nM T68251 CL1YO0 24954431 IC50 = 2.5 nM T68251 C3H9EO 24954432 IC50 = 7.6 nM T68251 CB60LR 24954795 IC50 = 24 nM T68251 C7P5YH 24954798 IC50 = 2.8 nM T68251 C5BG6I 24955154 IC50 = 32 nM T68251 CCE45B 24955155 IC50 = 56 nM T68251 CH53AG 24955156 IC50 = 47 nM T68251 CZC1P7 24955511 IC50 = 35 nM T68251 CL2G8J 24955513 IC50 = 281 nM T68251 CXG36M 24955514 IC50 = 4.8 nM T68251 CXO9Y4 24955857 IC50 = 36 nM T68251 CKY2F6 24955858 IC50 = 9.3 nM T68251 C4LJ8N 24955859 IC50 = 70 nM T68251 CX4MY3 24955861 IC50 = 67 nM T68251 CR29SO 24956227 IC50 = 509 nM T68251 CSM26P 24956228 IC50 = 102 nM T68251 C13JHO 24956229 IC50 = 4 nM T68251 C01QMC 24956580 IC50 = 1057 nM T68251 C8M5PJ 24956581 IC50 = 142 nM T68251 CC90AR 24956582 IC50 = 2382 nM T68251 CQH6I4 24956585 IC50 = 178 nM T68251 CHJ50Q 24956943 IC50 = 202 nM T68251 CN2AS5 24956945 IC50 = 670 nM T68251 C2HN8M 24956948 IC50 = 9.5 nM T68251 C2VEZ0 24957161 IC50 = 1318 nM T68251 CNCA57 25004194 Ki = 1.6 nM T68251 CIO26D 25022463 IC50 = 3 nM T68251 CWO3E0 25022465 IC50 = 170000 nM T68251 CAQ9Z1 25022681 Ki > 3333 nM T68251 CU6M9K 25060725 IC50 = 5400 nM T68251 CF7X2P 25060975 IC50 = 19000 nM T68251 CVR52U 25066764 IC50 = 60 nM T68251 CD2KA4 25102047 IC50 = 1.5 nM T68251 CRW96X 25102048 IC50 = 1 nM T68251 CQ3O9P 25102050 IC50 = 0.33 nM T68251 CSHA26 25102051 IC50 = 1.4 nM T68251 C7ADO2 25102197 IC50 = 0.37 nM T68251 CUR58H 25116339 IC50 = 297300 nM T68251 CA5DJ4 25138228 Ki = 2267000 nM T68251 CX6D9J 25138245 Ki > 3000 nM T68251 C7A6JQ 25138250 Ki = 5700 nM T68251 C6N7EQ 25138258 Ki > 3333 nM T68251 C7AD1J 25138259 Ki = 2933 nM T68251 CJ9TQ2 25138260 Ki > 3333 nM T68251 CUT8I7 25138261 Ki = 3300 nM T68251 CBD9X6 25138262 Ki > 3333 nM T68251 C8LX1S 25138263 Ki = 1367 nM T68251 C3OV1L 25138264 Ki > 3333 nM T68251 C92WVM 25138265 Ki > 3333 nM T68251 CMCS41 25138266 Ki > 3333 nM T68251 C1FJV5 25138267 Ki > 3333 nM T68251 C9N6WT 25138268 Ki > 3333 nM T68251 CF4QI1 25138269 Ki > 3333 nM T68251 C6P5UL 25138270 Ki > 3333 nM T68251 CQE0L7 25138271 Ki > 3333 nM T68251 C59XWU 25138272 Ki > 3333 nM T68251 C1TNQ3 25141117 Ki = 8.5 nM T68251 CYZ2J7 25141282 IC50 = 2 nM T68251 CR35QP 25144971 IC50 > 2500 nM T68251 C0Y5BC 25145683 IC50 > 2500 nM T68251 CGW49I 25146686 IC50 > 200000 nM T68251 CP0YF8 25146956 IC50 = 2900 nM T68251 C12AVL 25146957 IC50 = 3400 nM T68251 C10MBE 25146958 IC50 = 1500 nM T68251 CIUY75 25146959 IC50 = 2100 nM T68251 C5MG9N 25146960 IC50 = 6100 nM T68251 C83IOD 25147056 IC50 = 2200 nM T68251 C1IA0W 25147057 IC50 = 100 nM T68251 CB3W1I 25147058 IC50 = 800 nM T68251 CC35MZ 25147059 IC50 = 2200 nM T68251 CO5H9V 25147060 IC50 = 1600 nM T68251 CM20ZC 25147061 IC50 = 5 nM T68251 C2KZ0T 25147062 IC50 = 12 nM T68251 C5RMI2 25147153 IC50 = 100 nM T68251 C43YCQ 25147154 IC50 = 16 nM T68251 CPQW89 25147155 IC50 = 109 nM T68251 CQ3I6B 25147156 IC50 = 1100 nM T68251 CA34UT 25147158 IC50 = 4200 nM T68251 C3R0DB 25147159 IC50 = 5200 nM T68251 CV4ZE9 25147248 IC50 = 2100 nM T68251 C73HYI 25147249 IC50 = 3000 nM T68251 CV14TY 25147250 IC50 = 1 nM T68251 CUW8X2 25147251 IC50 = 4 nM T68251 C0Z7NX 25147252 IC50 = 11 nM T68251 CU1KO6 25147352 IC50 = 1000 nM T68251 CB1DY9 25147768 IC50 = 182900 nM T68251 CB7V8Y 25147773 IC50 = 0.35 nM T68251 C3KF1V 25178145 IC50 = 1.57 nM T68251 C8PMK7 25178356 IC50 > 100000 nM T68251 CG5Y2R 25178357 IC50 = 24.7 nM T68251 C4PZY6 25180866 IC50 = 145 nM T68251 CEP9Q2 25180867 IC50 = 0.5 nM T68251 C9HZG2 25181078 IC50 = 5120 nM T68251 CMYP34 25181079 IC50 = 2230 nM T68251 C7U1YC 25181080 IC50 = 25.3 nM T68251 C85HLG 25181081 IC50 = 16.2 nM T68251 CHR2P1 25183768 Ki > 25000 nM T68251 CZ8CR1 25190501 Ki > 3333 nM T68251 CO8CD1 25190502 Ki > 3333 nM T68251 C0R6MU 25212135 IC50 > 100000 nM T68251 C76PIF 26183540 IC50 = 33260 nM T68251 C9GCO4 28602444 IC50 = 48000 nM T68251 CW17CN 40516924 IC50 > 500000 nM T68251 C89YBJ 40582645 IC50 > 500000 nM T68251 C6AR8O 42623563 IC50 = 22000 nM T68251 CX0VP7 42623564 IC50 = 28000 nM T68251 C0H3RD 42627769 IC50 = 270 nM T68251 CB0QL3 42630085 IC50 = 37800 nM T68251 C7OX3C 42630086 IC50 = 47600 nM T68251 CAR56O 42645280 IC50 = 170200 nM T68251 CA6PS7 42645281 IC50 = 23500 nM T68251 C7R4JW 42645285 IC50 = 11200 nM T68251 CS29ZL 42645288 IC50 = 99700 nM T68251 C9JE0F 42645511 IC50 = 112100 nM T68251 CMK8T4 42645513 IC50 = 99700 nM T68251 CUF1L4 42645514 IC50 = 201900 nM T68251 C9WL3F 42645516 IC50 = 219400 nM T68251 C8OK0L 42645753 IC50 = 100700 nM T68251 C6K7LG 42645755 IC50 = 328500 nM T68251 CWS5M7 42645986 IC50 = 221000 nM T68251 CQBN65 42645987 IC50 = 632400 nM T68251 C6PI2X 42645989 IC50 = 211300 nM T68251 C8KM4E 43366432 IC50 = 8000 nM T68251 CPO1Z3 44123600 IC50 = 0.2 nM T68251 CWS64Q 44143474 IC50 > 15000 nM T68251 C7HV5Q 44143475 IC50 = 1590 nM T68251 C06IJY 44143476 IC50 = 1401 nM T68251 CVM82U 44143477 IC50 = 1241 nM T68251 C5XEB8 44143478 IC50 = 516 nM T68251 C0ZW7S 44143480 IC50 = 1093 nM T68251 C7K0YS 44143481 IC50 = 2674 nM T68251 CWU1K0 44143482 IC50 = 3614 nM T68251 CA29EQ 44143483 IC50 = 96 nM T68251 CA5P3E 44143484 IC50 = 15099 nM T68251 C7ER1N 44143485 IC50 = 855 nM T68251 C8YNO3 44143486 IC50 = 145 nM T68251 CLJG93 44143487 IC50 = 1743 nM T68251 CJB54F 44143488 IC50 = 2140 nM T68251 CH1IR0 44144307 IC50 = 14110 nM T68251 CT96JB 44199512 IC50 = 142900 nM T68251 C85BFQ 44199516 IC50 = 331100 nM T68251 CT80ED 44219901 Ki = 25 nM T68251 C94JVY 44219902 IC50 = 74 nM T68251 C7J6GH 44219903 IC50 = 26 nM T68251 C9J7WL 44219904 IC50 = 360 nM T68251 CRQ71E 44219905 IC50 = 310 nM T68251 C4Z0ID 44219906 IC50 = 56 nM T68251 CRNA25 44220092 IC50 = 17 nM T68251 C9T5ZF 44220093 IC50 = 9.6 nM T68251 CV38TE 44222825 IC50 = 5.5 nM T68251 CJI73R 44222826 IC50 = 1.5 nM T68251 CGQ30N 44222827 Ki = 3.8 nM T68251 CCI64J 44224245 IC50 = 66 nM T68251 CLRT69 44247751 IC50 = 3.5 nM T68251 CAR34Y 44263877 IC50 = 8.8 nM T68251 CEV08N 44263913 IC50 = 1.6 nM T68251 C5ZI0X 44263926 IC50 = 0.68 nM T68251 CO3C1E 44263994 IC50 = 2.7 nM T68251 C9XJ7U 44264020 IC50 = 3.4 nM T68251 C6L0MJ 44264021 IC50 = 2.4 nM T68251 CJ1WE7 44264036 IC50 = 0.7 nM T68251 C50QFR 44264375 IC50 = 5.3 nM T68251 CDL25C 44265349 Ki < 2.8 nM T68251 C3W4QO 44265401 Ki = 48 nM T68251 C2Q3JV 44265407 Ki = 2033 nM T68251 CN59QT 44265437 Ki = 500 nM T68251 CZA61K 44265475 Ki = 4.5 nM T68251 CD4A7F 44265476 Ki = 1133 nM T68251 CT6FK0 44265480 Ki < 2.8 nM T68251 C67HUL 44265485 Ki < 1 nM T68251 CH0O3I 44265492 Ki = 39 nM T68251 C4C7DY 44265493 Ki = 21 nM T68251 C0DFG7 44265501 Ki = 27 nM T68251 CXSD62 44265506 Ki = 310 nM T68251 CCM8K0 44265512 Ki = 2.8 nM T68251 CB3E6O 44265527 Ki < 2.8 nM T68251 COU3Y8 44266817 IC50 = 31 nM T68251 CUA5E0 44266818 IC50 = 8 nM T68251 CG23BI 44266830 IC50 = 8 nM T68251 C3YK0O 44268937 IC50 = 1000 nM T68251 C5DG8Z 44268941 IC50 = 200 nM T68251 C3SGT4 44268967 IC50 = 400 nM T68251 C1Z0GQ 44269012 IC50 = 1000 nM T68251 C18VGL 44269017 IC50 = 10000 nM T68251 CRF2Z5 44271421 IC50 = 8.05 nM T68251 CG7X5F 44272675 IC50 = 42.5 nM T68251 C2MWR0 44275913 Ki = 6.1 nM T68251 CKV1E7 44275972 Ki = 20 nM T68251 C6YT3K 44280285 Ki = 300 nM T68251 CC2O3U 44280323 Ki = 14 nM T68251 CIE09F 44280336 Ki = 0.3 nM T68251 CA1V6Y 44280345 Ki = 2 nM T68251 CI9L2E 44280411 Ki = 472 nM T68251 C8KZ2F 44281541 IC50 = 50 nM T68251 CRK8H6 44281557 IC50 = 66 nM T68251 CTJ7Q2 44281563 IC50 = 2.5 nM T68251 COU71D 44281564 IC50 = 64 nM T68251 CJ2PG9 44281705 IC50 = 23 nM T68251 C1M3JR 44281777 IC50 = 6.2 nM T68251 CL18QW 44281786 IC50 = 52 nM T68251 C3ES4Z 44281796 IC50 = 1.3 nM T68251 C60HIN 44281797 IC50 = 2.3 nM T68251 C8U5GR 44281941 IC50 = 110 nM T68251 CN23FC 44282968 IC50 = 1700 nM T68251 C2TV5I 44282969 IC50 = 50 nM T68251 CG3LF0 44282970 IC50 = 200 nM T68251 CC5XL3 44286083 IC50 = 48 nM T68251 CXT37W 44286406 IC50 = 35000 nM T68251 CB1R9G 44286414 IC50 > 10000 nM T68251 C7CU3J 44286466 IC50 = 19000 nM T68251 CZ2AL1 44286483 IC50 > 100000 nM T68251 C8I2EF 44286485 IC50 > 10000 nM T68251 C48FEB 44286518 IC50 = 130 nM T68251 CKM8V6 44286563 IC50 = 61 nM T68251 CJ1HT6 44288855 IC50 > 10000 nM T68251 CT38HI 44289140 IC50 > 10000 nM T68251 CAH30U 44289181 IC50 > 10000 nM T68251 CH1TS5 44289182 IC50 > 10000 nM T68251 CMZ2O6 44289200 IC50 > 10000 nM T68251 CBLC60 44289352 Ki = 31 nM T68251 CZO75J 44289369 Ki = 0.8 nM T68251 CRT7O2 44289382 Ki = 8 nM T68251 C7WUJ2 44289459 IC50 > 10000 nM T68251 CJ73FW 44289479 IC50 > 10000 nM T68251 CWMI67 44289482 IC50 > 10000 nM T68251 C1L4ZU 44289489 IC50 > 10000 nM T68251 C19EJM 44289515 IC50 > 10000 nM T68251 C6TI3X 44289520 Ki > 10000 nM T68251 CA52ED 44289521 Ki > 10000 nM T68251 C30KSP 44289579 Ki = 38 nM T68251 CHC08W 44289601 Ki = 36 nM T68251 CZ4EI7 44289602 Ki = 8 nM T68251 CEML82 44289603 Ki = 88 nM T68251 CM26JT 44289604 Ki = 27 nM T68251 CLY4K5 44289640 Ki = 4 nM T68251 C7GY8M 44289643 Ki > 10000 nM T68251 CV9B2F 44289867 Ki > 10000 nM T68251 CJ7VW3 44291166 IC50 = 0.7 nM T68251 C75IEN 44291420 IC50 = 30 nM T68251 CF21CS 44291532 IC50 = 0.7 nM T68251 CU75TB 44291559 IC50 = 53 nM T68251 C06JAO 44291626 IC50 = 49 nM T68251 C5XS0I 44294322 Ki = 1533 nM T68251 CC4V8S 44295180 IC50 = 50 nM T68251 CRW07Z 44295181 IC50 = 20 nM T68251 CL5QG6 44295202 IC50 = 540 nM T68251 CF0T8W 44295423 IC50 = 180 nM T68251 CVS7I1 44295425 IC50 = 550 nM T68251 CAFB18 44296974 Ki = 75 nM T68251 C5RSX9 44300181 IC50 = 19000 nM T68251 CKN3P7 44302022 IC50 = 100 nM T68251 C2Y0PK 44302023 IC50 = 9 nM T68251 C5S3UO 44302024 IC50 = 8 nM T68251 C8ERW6 44302042 IC50 = 10 nM T68251 C6JXH0 44302043 IC50 = 90 nM T68251 CI56DL 44302044 IC50 = 50 nM T68251 CWB83G 44302076 IC50 = 3 nM T68251 CY1J9U 44302096 IC50 = 5 nM T68251 CW94ZQ 44302164 IC50 = 47 nM T68251 C2FSR6 44302165 IC50 < 0.15 nM T68251 CQ54PZ 44302166 IC50 = 0.5 nM T68251 C9U3XT 44302167 IC50 = 0.6 nM T68251 C5X1WY 44302183 IC50 = 7 nM T68251 CQS19O 44302187 IC50 = 39810.72 nM T68251 C7G3BN 44302200 IC50 = 7 nM T68251 CMB4Q8 44302221 IC50 = 200 nM T68251 C70QWV 44302327 IC50 = 900 nM T68251 CZP20C 44302339 IC50 = 14 nM T68251 CO73BW 44302357 IC50 = 9 nM T68251 C6R0VK 44302358 IC50 = 500 nM T68251 CXUZ19 44302359 IC50 = 1 nM T68251 CNL4E2 44302361 IC50 = 19.95 nM T68251 C6YB0Q 44302364 IC50 = 10000 nM T68251 CCW65Y 44302378 IC50 = 1.995 nM T68251 CDK9W1 44302383 IC50 = 30.2 nM T68251 CYG80V 44302385 IC50 = 15 nM T68251 C7ZBR4 44302396 IC50 = 0.6 nM T68251 C8S5WT 44302397 IC50 = 1 nM T68251 CPC25G 44302409 IC50 = 13 nM T68251 C4QL0I 44302411 IC50 = 1 nM T68251 C4NDA2 44302416 IC50 = 12 nM T68251 C24ZWF 44302429 IC50 = 17 nM T68251 C4I6WO 44302430 IC50 = 0.8 nM T68251 CYL71W 44302432 IC50 = 3 nM T68251 C2X3QG 44302433 IC50 = 1000 nM T68251 C1J2AN 44302479 IC50 = 794.33 nM T68251 CE3BX0 44302505 IC50 = 200 nM T68251 C5H6OV 44302627 IC50 = 8 nM T68251 C6QR7C 44302634 IC50 = 15 nM T68251 CG8KJ0 44302661 IC50 = 5 nM T68251 CUZS20 44302663 IC50 = 600 nM T68251 CX1M3Q 44302666 IC50 = 6 nM T68251 C36CQP 44302952 IC50 = 12 nM T68251 CALD50 44304020 Ki > 3000 nM T68251 CTU4S6 44304048 Ki > 3000 nM T68251 CSVK45 44304230 Ki > 3000 nM T68251 CLH14M 44305978 IC50 = 5.9 nM T68251 CZ49UN 44305988 IC50 = 2.3 nM T68251 C6I8JA 44306058 IC50 = 1.9 nM T68251 CB5EY3 44306200 IC50 = 6.5 nM T68251 C0YOH1 44306202 IC50 = 3.8 nM T68251 CMA39E 44306203 IC50 = 2.1 nM T68251 CL58OS 44306208 IC50 = 14000 nM T68251 CAY2S4 44306209 IC50 = 1400 nM T68251 C27NJX 44306277 IC50 = 0.3 nM T68251 C6O1AN 44306279 IC50 = 0.8 nM T68251 C5AM6P 44308844 IC50 = 1587.17 nM T68251 CZUY51 44310789 Ki = 8.1 nM T68251 CH92OI 44310813 Ki = 3 nM T68251 CI4Y5N 44310825 Ki = 13 nM T68251 C5W8QH 44310847 Ki = 6.9 nM T68251 CLQV12 44310863 Ki = 0.44 nM T68251 CN9P5A 44310921 Ki = 0.42 nM T68251 CXB76U 44310932 Ki = 0.7 nM T68251 CMW5G3 44310933 Ki = 8.1 nM T68251 CBY0T1 44310973 Ki = 25 nM T68251 C5D9FS 44311011 Ki = 0.59 nM T68251 C2GC9W 44311172 Ki = 18 nM T68251 C0K1IL 44311187 Ki = 1.3 nM T68251 CL3CS0 44311254 Ki = 43 nM T68251 CV63JP 44311265 Ki = 1.9 nM T68251 CS56ER 44311267 Ki = 46 nM T68251 C5MBT7 44311268 Ki = 7.5 nM T68251 CM64HK 44311313 Ki = 1.9 nM T68251 CLQ48B 44311332 Ki = 6.7 nM T68251 C5AO7Z 44311335 Ki = 0.7 nM T68251 C78TEU 44311349 Ki = 0.96 nM T68251 CJEM64 44311491 Ki = 1.1 nM T68251 C2W5NQ 44311510 Ki = 0.47 nM T68251 C2MIT8 44311525 Ki = 1 nM T68251 CP7L6Q 44311566 Ki = 4 nM T68251 C0B4HZ 44312333 Ki = 12.88 nM T68251 CK9XB7 44314087 IC50 = 20 nM T68251 C8MRB1 44314322 IC50 = 0.36 nM T68251 CB6UL7 44314349 IC50 = 1.5 nM T68251 C3R0DL 44314366 IC50 = 1.9 nM T68251 C5ZTU6 44314442 Ki = 3.82 nM T68251 C2JUX9 44314443 Ki = 1.17 nM T68251 C92MGV 44314566 IC50 = 0.86 nM T68251 CLT6E0 44314618 IC50 = 3.7 nM T68251 CC95EZ 44314744 Ki = 0.33 nM T68251 CY63DG 44314754 Ki = 0.01 nM T68251 C8ZD7F 44314755 Ki = 10 nM T68251 COF0B1 44314762 Ki = 0.08 nM T68251 C59CBZ 44314763 Ki = 0.06 nM T68251 C9L1NY 44314788 Ki = 0.01 nM T68251 CM04TG 44314789 Ki = 0.03 nM T68251 C7LCN0 44314824 Ki = 10.3 nM T68251 CNM6W8 44314841 Ki = 0.01 nM T68251 C9K8JZ 44314900 Ki = 0.254 nM T68251 CXRE70 44314901 Ki = 0.06 nM T68251 CK3H1Y 44314929 Ki = 2.24 nM T68251 CS5A6Z 44314930 Ki = 0.06 nM T68251 CNB72W 44314931 Ki = 0.05 nM T68251 CBXI30 44314932 Ki = 0.02 nM T68251 CCF80X 44314958 Ki = 812 nM T68251 C3N8RQ 44314969 Ki = 1.83 nM T68251 C9SRT4 44314970 Ki = 1.03 nM T68251 C61DST 44314974 Ki = 0.03 nM T68251 CE2J4M 44314975 Ki = 0.01 nM T68251 CQE0D3 44314976 Ki = 0.59 nM T68251 CI2V1Y 44314995 Ki = 123 nM T68251 C48NVD 44314999 Ki = 0.01 nM T68251 CB7F0J 44315000 Ki = 0.3 nM T68251 CSY78M 44315028 Ki = 1300 nM T68251 CDZ5O3 44315029 Ki = 550 nM T68251 C6HW5G 44315084 Ki = 0.01 nM T68251 CV6KW1 44315085 Ki = 0.02 nM T68251 CH48TD 44315155 IC50 = 110 nM T68251 CAUQ47 44315167 Ki = 6 nM T68251 COA01P 44315179 Ki = 3000 nM T68251 CQ1R9E 44315204 Ki = 3.06 nM T68251 CL32FZ 44315221 Ki = 620 nM T68251 CDN4Y5 44315222 Ki = 860 nM T68251 C62FXJ 44315244 IC50 = 2.6 nM T68251 CP9M6W 44315277 Ki = 0.1 nM T68251 C3SZO4 44315279 Ki = 18.9 nM T68251 CSG05N 44315321 Ki = 0.02 nM T68251 COD08C 44315324 Ki = 46.5 nM T68251 C50IQE 44315333 IC50 = 6.6 nM T68251 C37JMW 44315348 Ki = 6.4 nM T68251 C89IQW 44318090 IC50 = 1 nM T68251 CJU31O 44321285 Ki = 17 nM T68251 C41VFA 44321286 Ki = 8 nM T68251 C5S2ZU 44321484 Ki = 85 nM T68251 CLQ23M 44321485 Ki = 202 nM T68251 CHF76Q 44321540 Ki = 9 nM T68251 CVOL49 44321593 Ki = 30 nM T68251 CB97GK 44321601 Ki = 26 nM T68251 CT0O7Y 44321602 Ki = 260 nM T68251 CU62BP 44321746 Ki = 11 nM T68251 CQU2K9 44321782 Ki = 100 nM T68251 CV8T3N 44321783 Ki = 19 nM T68251 CIBO50 44321801 Ki = 6 nM T68251 C4E8GU 44321802 Ki = 30 nM T68251 CYDN18 44321803 Ki = 40 nM T68251 C7Z4DQ 44321887 Ki = 24 nM T68251 CFJ20T 44321932 Ki = 10 nM T68251 C2E3RF 44321966 Ki = 75 nM T68251 CW9S1N 44321967 Ki = 330 nM T68251 C1FI3O 44321975 Ki = 14 nM T68251 CLB8J6 44321976 Ki = 80 nM T68251 CR0KN1 44322209 Ki = 250 nM T68251 C5LE1P 44322210 Ki = 31 nM T68251 CQ7AW8 44322211 Ki = 250 nM T68251 CJY2O7 44322214 Ki = 275 nM T68251 CR9GI0 44322215 Ki = 145 nM T68251 CYR6E5 44323170 Ki = 2000 nM T68251 C29OCD 44325165 Ki = 90 nM T68251 C20UGO 44325517 Ki = 157 nM T68251 C1SRC9 44325555 Ki = 6.9 nM T68251 CHMC02 44325564 Ki = 210 nM T68251 C8P6UA 44325625 Ki = 0.02 nM T68251 CBY75J 44325686 Ki = 1900 nM T68251 C6A1JX 44325696 Ki = 0.05 nM T68251 CJU3R8 44325730 Ki = 0.01 nM T68251 CBV73K 44325744 Ki = 0.03 nM T68251 C06ZAH 44325745 Ki = 0.01 nM T68251 C70UFH 44325749 Ki = 0.02 nM T68251 C8EWP2 44325750 Ki = 0.02 nM T68251 C2QL0B 44325810 Ki = 0.03 nM T68251 CS4EV5 44325831 IC50 = 3000 nM T68251 CU9B2Q 44325832 IC50 = 220 nM T68251 CP1NU9 44325834 Ki = 0.59 nM T68251 C7VRX2 44325907 Ki = 0.01 nM T68251 C80RKL 44326171 IC50 > 100000 nM T68251 C64XEI 44326172 IC50 = 670 nM T68251 C08MOK 44326187 IC50 > 100000 nM T68251 C3UB9D 44326260 IC50 = 17000 nM T68251 C1D8RA 44326261 IC50 = 2000 nM T68251 CK6P3C 44326668 IC50 = 370 nM T68251 C63XAO 44327476 IC50 = 90000 nM T68251 C7S4GH 44327780 IC50 = 200000 nM T68251 CXO1S8 44327801 IC50 = 100000 nM T68251 CW1QN6 44327818 IC50 > 500000 nM T68251 CTH2Y7 44327914 IC50 = 120000 nM T68251 CWYJ75 44327915 IC50 = 150000 nM T68251 C27ZST 44327916 IC50 = 60000 nM T68251 COAF26 44327936 IC50 > 500000 nM T68251 C9O8LM 44327939 IC50 = 160000 nM T68251 CB5L2U 44327940 IC50 = 72000 nM T68251 CI29FZ 44327960 IC50 = 155000 nM T68251 CV2U6R 44327961 IC50 = 54000 nM T68251 C8HUF1 44328149 IC50 > 500000 nM T68251 C85QTP 44328155 IC50 = 1000 nM T68251 CLK87J 44328168 IC50 = 150000 nM T68251 CMHZ13 44328169 IC50 > 500000 nM T68251 CZQ6N7 44328189 IC50 > 100000 nM T68251 C1IG0A 44328244 IC50 = 230000 nM T68251 CEI1V4 44328245 IC50 = 40000 nM T68251 CPI3A5 44328246 IC50 = 100000 nM T68251 CPU60Z 44328254 IC50 = 150000 nM T68251 CW3RX8 44328256 IC50 = 370000 nM T68251 CN81EA 44328258 IC50 = 43000 nM T68251 CR8XQ3 44328259 IC50 = 114000 nM T68251 CCD48V 44328263 IC50 = 2000 nM T68251 C31OKH 44328271 IC50 > 500000 nM T68251 CUA04P 44328279 IC50 = 125000 nM T68251 CHB05O 44328283 IC50 = 52000 nM T68251 CLC39W 44328295 IC50 = 110000 nM T68251 C36FCK 44328296 IC50 = 51000 nM T68251 CI46AP 44328297 IC50 > 500000 nM T68251 CR9YN5 44328312 IC50 > 500000 nM T68251 C8W9KN 44328316 IC50 = 50000 nM T68251 CPT80U 44328317 IC50 = 60000 nM T68251 CBD0Z2 44329014 IC50 = 5.97 nM T68251 CMLA39 44329018 IC50 = 1.3 nM T68251 C84MVU 44329019 IC50 = 5.73 nM T68251 C90CHA 44329405 IC50 = 7079.46 nM T68251 C2PB4Z 44329622 IC50 = 500 nM T68251 CI3Z4K 44329623 IC50 = 80 nM T68251 C6OL8M 44329636 IC50 = 10000 nM T68251 CB0G1H 44329644 IC50 = 1995.26 nM T68251 CA65RO 44329672 IC50 = 1995.26 nM T68251 CK9HO7 44329673 IC50 = 2000 nM T68251 C07GRS 44329693 IC50 = 60 nM T68251 CBH16R 44329694 IC50 = 600 nM T68251 CG3E7A 44329712 IC50 = 19.95 nM T68251 C9SN6I 44329713 IC50 = 3000 nM T68251 CZ2FW6 44329725 IC50 = 1995.26 nM T68251 CDKI48 44329741 IC50 = 500 nM T68251 CK3M2H 44329742 IC50 = 3000 nM T68251 C39RDS 44329886 IC50 = 50 nM T68251 C3YAF6 44329898 IC50 = 7000 nM T68251 C63RHP 44329909 IC50 = 95.5 nM T68251 CVQA75 44329910 IC50 = 398.11 nM T68251 C84SLI 44329926 IC50 = 100 nM T68251 CJS6B1 44329927 IC50 = 398.11 nM T68251 C2K6OU 44329943 IC50 = 95.5 nM T68251 C5BYR4 44329998 IC50 = 3400 nM T68251 C0SMC9 44330092 IC50 = 21 nM T68251 C35SIO 44330094 IC50 = 12.88 nM T68251 C3NM2G 44330095 IC50 = 0.7943 nM T68251 C6SCU5 44330119 IC50 = 0.26 nM T68251 C69KPL 44330130 IC50 = 109.65 nM T68251 C9P6ZF 44330131 IC50 = 10 nM T68251 C9R1ZE 44330132 IC50 = 55000 nM T68251 CKS01F 44330133 IC50 = 2187.76 nM T68251 CLU8I7 44330135 IC50 = 7000 nM T68251 C1IE0S 44330147 IC50 > 100000 nM T68251 CPG7N2 44330149 IC50 = 15000 nM T68251 CYP6S4 44330152 IC50 = 6000 nM T68251 CMGA28 44330163 IC50 = 41000 nM T68251 CXI49L 44330197 IC50 = 4000 nM T68251 CDQM84 44330198 IC50 = 0.048 nM T68251 CH6EN4 44330225 IC50 = 3388.44 nM T68251 C3GA9Q 44330226 IC50 = 0.23 nM T68251 CG2Q8W 44332306 IC50 = 36 nM T68251 C5NG0R 44334948 IC50 = 30 nM T68251 CFP3X8 44334949 IC50 = 53 nM T68251 CV5RF0 44334963 IC50 = 441 nM T68251 C4AOZ7 44334981 IC50 = 143 nM T68251 CXW59C 44334982 IC50 = 4.6 nM T68251 CCH1W8 44334983 IC50 = 2.5 nM T68251 CQ0UI1 44335017 IC50 = 32 nM T68251 CX58SB 44335240 IC50 = 1.64 nM T68251 CA96JG 44335285 IC50 = 15.4 nM T68251 CI5X0G 44339523 IC50 = 7.2 nM T68251 CB9K8T 44339536 IC50 = 9.5 nM T68251 C2R3XN 44339554 IC50 = 6.5 nM T68251 C2CRY1 44339556 IC50 = 8.6 nM T68251 CTBU53 44339564 IC50 = 23 nM T68251 C58OSK 44339567 IC50 = 7.2 nM T68251 CX2KJ3 44339574 IC50 = 110 nM T68251 CEK3G0 44339588 IC50 = 8.5 nM T68251 C7ZR6H 44339589 IC50 = 1100 nM T68251 C0WP9C 44339590 IC50 = 2.7 nM T68251 C5C2LI 44339654 IC50 = 1 nM T68251 CLD2P9 44339900 Ki = 4400 nM T68251 C2D6VN 44339918 Ki = 2.1 nM T68251 CRQJ09 44339936 Ki = 1300 nM T68251 C4JLG8 44340091 Ki = 6.1 nM T68251 CXW34P 44340094 Ki = 19 nM T68251 CGV94P 44340160 Ki = 7.3 nM T68251 C3IS1O 44340161 Ki = 130 nM T68251 CPK5W0 44340172 Ki = 26 nM T68251 CJ4Z9W 44340207 Ki = 570 nM T68251 CZ31VY 44340208 Ki = 12 nM T68251 C4B9QZ 44340327 Ki = 20 nM T68251 C2XY8H 44340328 Ki = 2.1 nM T68251 CAT48Z 44340657 Ki = 20 nM T68251 C3CYZ8 44340673 Ki = 1100 nM T68251 CRI8Q4 44340696 Ki = 1100 nM T68251 CF1QZ3 44340718 Ki = 70 nM T68251 C09ILT 44340727 Ki = 120 nM T68251 C6AS8J 44340740 Ki = 570 nM T68251 CL0U9T 44340810 Ki = 60 nM T68251 CV6W7Z 44340812 Ki = 770 nM T68251 C3WZM0 44340828 Ki = 2300 nM T68251 CW53EF 44340868 Ki = 350 nM T68251 C6ZDV3 44340869 Ki = 120 nM T68251 CR1ID4 44340923 Ki = 110 nM T68251 CL9I4M 44341538 Ki = 1533 nM T68251 CE3MT4 44341611 Ki = 4650 nM T68251 CJTZ45 44341652 Ki = 200000 nM T68251 C2XP4N 44342352 Ki = 3000 nM T68251 C2SZB1 44342614 IC50 = 6 nM T68251 CTQ6P4 44344631 IC50 = 34200 nM T68251 CBH9I5 44344658 IC50 = 750 nM T68251 CCF94Z 44349787 IC50 = 572 nM T68251 C1L2GF 44350073 IC50 = 20 nM T68251 CQ5RN6 44350101 IC50 = 130 nM T68251 CE2X3Q 44350116 IC50 > 100 nM T68251 CO9R4W 44356376 Ki > 3333 nM T68251 C3MZA1 44356386 Ki > 3333 nM T68251 CH1E2S 44356406 Ki > 3333 nM T68251 C84LUM 44356631 Ki > 3333 nM T68251 CG6T9A 44356632 Ki > 3333 nM T68251 C3WFH7 44356634 Ki > 3333 nM T68251 CB8KY4 44356635 Ki > 3333 nM T68251 COIA82 44356636 Ki > 3333 nM T68251 C4BU6T 44356644 Ki > 3333 nM T68251 CH9YT4 44356659 Ki > 3333 nM T68251 C68LMR 44356675 Ki > 3333 nM T68251 C69YIP 44356686 Ki > 3333 nM T68251 CT05XN 44356687 Ki 1079 nM T68251 CML03W 44356689 Ki > 3333 nM T68251 CQ4NP5 44356690 Ki > 3333 nM T68251 CE8U2Y 44356714 Ki > 3333 nM T68251 CCY5U3 44356804 Ki = 200 nM T68251 C27LMU 44356852 Ki > 3333 nM T68251 CTU64D 44356889 Ki > 3333 nM T68251 C4TM1I 44356890 Ki > 3333 nM T68251 C1WA4B 44356906 Ki > 3333 nM T68251 C50ELY 44356907 Ki 675 nM T68251 CVU8L2 44356924 Ki > 3333 nM T68251 CD1GW2 44356953 Ki > 1011 nM T68251 CR41QN 44356969 Ki > 2454 nM T68251 C3BT0N 44356971 Ki = 642 nM T68251 C81OIZ 44356983 Ki > 3333 nM T68251 CHNC03 44356993 Ki > 3333 nM T68251 C9Z3RT 44356998 Ki > 3333 nM T68251 CR4A7G 44356999 Ki = 476 nM T68251 C2VS6P 44357000 Ki = 1537 nM T68251 CES1G8 44357007 Ki > 3333 nM T68251 C6NQ7K 44357012 Ki = 656 nM T68251 C2HIN3 44357023 Ki > 3333 nM T68251 CI4JO7 44357024 Ki 585 nM T68251 CW4VQ3 44357029 Ki > 3333 nM T68251 C2AIT6 44357209 Ki > 3333 nM T68251 CJK2P7 44357220 Ki > 3333 nM T68251 CIX6G5 44357225 Ki > 3333 nM T68251 CT4C6P 44360260 IC50 = 4.2 nM T68251 CY5I3O 44360286 IC50 = 35 nM T68251 C40OCB 44360287 IC50 = 1.8 nM T68251 C3IW9L 44360784 IC50 = 1.4 nM T68251 CGQ92A 44364037 IC50 = 33 nM T68251 C36YLM 44364111 IC50 = 150 nM T68251 CN4T7Q 44364119 IC50 = 76 nM T68251 CH4TE7 44364121 IC50 = 24 nM T68251 CPE91Y 44364122 IC50 = 18 nM T68251 CG2X0C 44364224 IC50 = 430 nM T68251 C1F8XN 44364249 IC50 = 26 nM T68251 CWM47H 44364250 IC50 = 27 nM T68251 C0W5TL 44364251 IC50 = 1099 nM T68251 C3TPO7 44364266 IC50 = 853 nM T68251 CJ2B8F 44364280 IC50 = 724 nM T68251 C90CYD 44367175 IC50 = 4 nM T68251 C2DV0R 44367276 IC50 = 0.5 nM T68251 C5BAW2 44367284 IC50 < 0.4 nM T68251 C2YG5E 44367285 IC50 = 11 nM T68251 CUDF82 44367309 IC50 = 1 nM T68251 CA0CJ1 44368580 IC50 = 25.7 nM T68251 CW0Y3K 44368632 IC50 = 30 nM T68251 CU8FD2 44368650 IC50 = 109.65 nM T68251 CLE71V 44368654 IC50 = 15.14 nM T68251 CQ27XL 44368655 IC50 = 3.388 nM T68251 CH9G3O 44368849 IC50 = 1 nM T68251 CV6ZG4 44368850 IC50 = 1.288 nM T68251 CB2U9G 44368858 IC50 = 270 nM T68251 CN78UB 44368864 IC50 = 5.754 nM T68251 CV8ZA4 44368865 IC50 = 1.585 nM T68251 CW8O3S 44368924 IC50 = 50.12 nM T68251 C6CD9A 44368928 IC50 = 280 nM T68251 C5HF6P 44368940 IC50 = 330 nM T68251 CE30XV 44368941 IC50 = 50 nM T68251 CG2P9T 44368942 IC50 = 83.18 nM T68251 C7HT1U 44368944 IC50 = 3467.37 nM T68251 C1CW5A 44368946 IC50 = 6165.95 nM T68251 CV86QS 44368963 IC50 = 331.13 nM T68251 C4C7UJ 44368968 IC50 = 38 nM T68251 C3EW6B 44368969 IC50 = 416.87 nM T68251 C4I6ME 44368970 IC50 = 61 nM T68251 C8IZC4 44369030 IC50 = 2430 nM T68251 CDW8V9 44369031 IC50 = 6.4 nM T68251 C82BOI 44369038 IC50 = 776.25 nM T68251 C65FBJ 44369041 IC50 = 53.7 nM T68251 CI0S2R 44369094 IC50 = 310 nM T68251 CFI10T 44369095 IC50 = 34 nM T68251 CQGM80 44369096 IC50 = 210 nM T68251 CIR84S 44369104 IC50 = 920 nM T68251 C6SBW5 44369107 IC50 = 100 nM T68251 CAF5P0 44369163 IC50 = 52000 nM T68251 CHC71X 44369164 IC50 = 1700 nM T68251 CY5L0D 44369186 IC50 = 1 nM T68251 C1JZK6 44369209 IC50 = 86 nM T68251 C9BAO2 44369213 IC50 = 6800 nM T68251 CCJ63B 44369214 IC50 = 11 nM T68251 C4E7DM 44369266 IC50 = 41 nM T68251 CI0ZD9 44371783 IC50 = 20 nM T68251 C4VR5M 44371799 IC50 = 251 nM T68251 C4FHG7 44371800 IC50 = 38 nM T68251 CQ5UR4 44372530 IC50 = 240 nM T68251 CCZ6J3 44379232 Ki = 470 nM T68251 CW20ML 44379249 Ki = 110 nM T68251 CXM06G 44379250 Ki = 5.7 nM T68251 CK0B1D 44379273 Ki = 220 nM T68251 COD6P1 44379499 Ki = 2.6 nM T68251 C84YPO 44379547 Ki > 1000 nM T68251 C3EV2A 44384940 IC50 = 530 nM T68251 C0XE8K 44384941 IC50 = 13000 nM T68251 C3IJO9 44384994 IC50 > 50000 nM T68251 CZ6PU7 44389401 Ki = 1.8 nM T68251 CO4W0Y 44389552 Ki = 0.4 nM T68251 CWQ19I 44389560 IC50 = 10.3 nM T68251 C5R4EW 44389591 IC50 = 935 nM T68251 CC7QW9 44391352 IC50 = 21 nM T68251 C89FTQ 44393434 Ki > 3300 nM T68251 CCO3S9 44393444 Ki > 3300 nM T68251 CNO4P6 44393516 Ki > 3300 nM T68251 C5OIK4 44393520 Ki > 3300 nM T68251 C80NZE 44394179 Ki > 3300 nM T68251 CXD05N 44394645 Ki > 100000 nM T68251 CGQ98X 44394681 Ki = 153000 nM T68251 C8MY4S 44394703 Ki = 88000 nM T68251 CCEI41 44394814 Ki > 2000000 nM T68251 CCZ09V 44394886 Ki > 100000 nM T68251 CZB81D 44395506 IC50 = 5 nM T68251 CAU5R4 44397021 IC50 = 23.3 nM T68251 CQR73V 44397047 IC50 = 27.8 nM T68251 CSO92L 44397377 IC50 = 1.9 nM T68251 CMWU78 44397457 IC50 = 19 nM T68251 CU1E2Z 44397536 IC50 = 14 nM T68251 CQ1Y4E 44397568 IC50 = 4 nM T68251 C12MNT 44397632 IC50 = 2 nM T68251 CZ45GV 44397680 IC50 = 12.1 nM T68251 C7Y1VK 44397699 IC50 = 3.9 nM T68251 CHL9S2 44399294 Ki = 2530 nM T68251 CD49UI 44399312 Ki = 600 nM T68251 C3LS8N 44399509 Ki = 3330 nM T68251 CIA8T3 44399555 Ki > 3330 nM T68251 C8PR7S 44400182 IC50 = 9 nM T68251 CQ9F0K 44400232 IC50 = 9 nM T68251 C91POV 44402021 IC50 = 197 nM T68251 CYCJ78 44402280 IC50 = 9.8 nM T68251 CWG3M4 44402281 IC50 > 10000 nM T68251 C9KGL0 44404474 IC50 = 0.91 nM T68251 C92KDG 44404475 IC50 = 7.1 nM T68251 C07CGB 44404477 IC50 = 1050 nM T68251 C7VH3G 44404484 IC50 = 259 nM T68251 CC29XL 44404490 IC50 = 1770 nM T68251 CCN16G 44404500 IC50 = 164 nM T68251 C69GZU 44404501 IC50 = 688 nM T68251 CY6WL5 44404502 IC50 = 1490 nM T68251 CWGQ46 44404503 IC50 = 1610 nM T68251 CLXM58 44404504 IC50 = 2500 nM T68251 C1F9HO 44404506 IC50 = 4340 nM T68251 CLU41O 44404507 IC50 = 7000 nM T68251 C30DKN 44404553 IC50 = 0.04 nM T68251 C0G4MR 44405997 IC50 > 380000 nM T68251 CZ0XC1 44405998 IC50 = 685000 nM T68251 CIC60V 44406452 IC50 = 28 nM T68251 CHM26J 44406652 Ki = 8100 nM T68251 C1K3QM 44406655 IC50 = 20 nM T68251 C6YG5S 44406678 IC50 = 2.6 nM T68251 CB5ZS0 44411587 IC50 = 52 nM T68251 C4Z0BX 44411591 IC50 = 3060 nM T68251 CHV64P 44411592 IC50 = 0.84 nM T68251 CL6IG9 44411599 IC50 = 6.8 nM T68251 C6IKL1 44411602 IC50 = 0.7 nM T68251 CM2UL0 44411603 IC50 = 1.5 nM T68251 CBT4E7 44411614 IC50 = 4 nM T68251 CH8B4W 44411639 IC50 = 1.1 nM T68251 CS74LI 44411640 IC50 = 54 nM T68251 C43HTC 44411693 IC50 = 3 nM T68251 C8HSN2 44411697 IC50 = 1.2 nM T68251 CKQ8P6 44411698 IC50 = 0.74 nM T68251 CVQ82B 44411701 IC50 = 33 nM T68251 C87VNZ 44411702 IC50 = 1.3 nM T68251 C83MTG 44411776 IC50 = 0.98 nM T68251 CT1A8Q 44411815 IC50 = 295 nM T68251 CQLV08 44411816 IC50 = 556 nM T68251 CP16XL 44411819 IC50 = 1.8 nM T68251 C9COT4 44411820 IC50 = 6.5 nM T68251 C3Q8PM 44411822 IC50 = 4.4 nM T68251 CEB0S4 44411823 IC50 = 0.7 nM T68251 CRB85W 44411826 IC50 = 2.3 nM T68251 CV1NO8 44411829 IC50 = 1.7 nM T68251 CPH6V5 44411830 IC50 = 0.62 nM T68251 CRKL06 44411835 IC50 = 145 nM T68251 C0FDM1 44411836 IC50 = 8.6 nM T68251 CUV27I 44411839 IC50 = 19 nM T68251 CD5KV9 44411846 IC50 = 12 nM T68251 C7CU1F 44411852 IC50 = 1.3 nM T68251 CA9OS4 44411865 IC50 = 1.9 nM T68251 CVM7Y3 44413975 IC50 = 49 nM T68251 C4X0GA 44413977 IC50 = 15 nM T68251 CH01EO 44413978 IC50 = 24 nM T68251 CQ8HK9 44413979 IC50 = 553 nM T68251 CBT0P2 44413982 IC50 = 46 nM T68251 CIJ39D 44413983 IC50 = 16 nM T68251 C9BA0V 44413987 IC50 = 111 nM T68251 CE3WP0 44413991 IC50 = 518 nM T68251 CDUI73 44413992 IC50 = 3.1 nM T68251 CH2X6W 44413997 IC50 = 44 nM T68251 CHN85S 44414002 IC50 = 345 nM T68251 C2OJ4B 44414029 IC50 = 302 nM T68251 CT5PC9 44422672 IC50 = 2.3 nM T68251 CS9D5U 44422720 IC50 = 0.39 nM T68251 CNWM05 44422723 IC50 = 1.8 nM T68251 C58LAY 44422724 IC50 = 20 nM T68251 CDQU41 44422736 IC50 = 53 nM T68251 CVUB56 44422737 IC50 = 30 nM T68251 CB8G2W 44422743 IC50 = 24 nM T68251 CFX42T 44422744 IC50 = 980 nM T68251 C9EL7F 44422749 IC50 = 790 nM T68251 CY49HT 44423674 IC50 = 9600 nM T68251 CHI5G1 44423675 IC50 = 1060 nM T68251 CFC3M6 44423676 IC50 = 1500 nM T68251 CO24JF 44423677 IC50 = 5000 nM T68251 C7F9DB 44423678 IC50 = 30000 nM T68251 CJ6GW5 44423679 IC50 = 1980 nM T68251 CUKM29 44423680 IC50 = 2100 nM T68251 C3R0FS 44423681 IC50 = 660 nM T68251 C14DBJ 44423682 IC50 = 730 nM T68251 CU5QV9 44425142 IC50 > 100000 nM T68251 CW8RY1 44425150 IC50 = 5900 nM T68251 C45WZX 44426073 IC50 = 10 ug.mL-1 T68251 CK5H7O 44429877 IC50 = 5000 nM T68251 CQL1X9 44429878 IC50 = 73 nM T68251 C1CYV2 44429879 IC50 = 82 nM T68251 C7AXP9 44429880 IC50 = 58 nM T68251 CXOS97 44429881 IC50 = 11 nM T68251 C2MQ0I 44429882 IC50 = 37 nM T68251 CQ5PT8 44429883 IC50 = 37 nM T68251 CQRO36 44429884 IC50 = 161 nM T68251 CM27YB 44429885 IC50 = 54 nM T68251 C9JH0T 44429886 IC50 = 4 nM T68251 CD2B3T 44429887 IC50 = 62.6 nM T68251 C6V1CO 44429888 IC50 = 2058 nM T68251 CBC6W4 44429889 IC50 = 40 nM T68251 C7A0LF 44429890 IC50 = 176 nM T68251 CS0M3L 44429891 IC50 = 99.5 nM T68251 CX93QY 44429892 IC50 = 19 nM T68251 C7SWV1 44429893 IC50 = 33 nM T68251 C8QKS0 44429894 IC50 = 22 nM T68251 CBS47K 44429896 IC50 = 32 nM T68251 CI7TG1 44429897 IC50 = 61.3 nM T68251 CLJ48T 44429898 IC50 = 51 nM T68251 C3F9CK 44429899 IC50 = 51 nM T68251 C8PVF7 44429900 IC50 = 31 nM T68251 C6U0TK 44429901 IC50 = 20 nM T68251 CBK9M5 44429902 IC50 = 58 nM T68251 C72YFT 44429903 IC50 = 172 nM T68251 CMO9Q3 44429905 IC50 = 183 nM T68251 C8BHL5 44431844 IC50 > 2000 nM T68251 CR1DN9 44431845 IC50 > 2000 nM T68251 CHFB16 44431846 IC50 > 2000 nM T68251 C0C3ZT 44431847 IC50 > 2000 nM T68251 CS49GV 44431848 IC50 > 2000 nM T68251 C4AVK5 44431849 IC50 > 2000 nM T68251 C5DH4Q 44431850 IC50 > 2000 nM T68251 CLHE45 44431851 IC50 > 2000 nM T68251 CYG29L 44431852 IC50 > 2000 nM T68251 C4OF5L 44431853 IC50 > 2000 nM T68251 CWU7G8 44434565 IC50 = 123 nM T68251 CF9HU5 44434566 IC50 = 280 nM T68251 CV3M6F 44434578 IC50 = 120 nM T68251 CJN1K9 44439853 Ki = 20 nM T68251 C71IPQ 44439982 IC50 = 4000 nM T68251 C2WJP3 44439983 IC50 = 4400 nM T68251 CU9Z1H 44439984 IC50 = 1000 nM T68251 C0G4AS 44439985 IC50 = 3800 nM T68251 CV8D9L 44439986 IC50 = 4300 nM T68251 CKP8T1 44439987 IC50 = 2200 nM T68251 CUT86C 44439988 IC50 = 1200 nM T68251 CKC81R 44439990 IC50 = 1200 nM T68251 CPNM45 44439991 IC50 = 600 nM T68251 CROG92 44439992 IC50 = 300 nM T68251 C30RNZ 44439993 IC50 = 1200 nM T68251 C19MPB 44439994 IC50 = 13000 nM T68251 C2N1UC 44439995 IC50 = 1400 nM T68251 C4T0AW 44439996 IC50 = 1800 nM T68251 CJT4H2 44439997 IC50 = 1300 nM T68251 CYM08I 44439998 IC50 = 1700 nM T68251 C83KQO 44439999 IC50 = 15600 nM T68251 C4Y9JD 44440000 IC50 = 500 nM T68251 C5PWG9 44440001 IC50 = 10600 nM T68251 C70MGQ 44440455 Ki > 3333 nM T68251 CDY53F 44440460 Ki > 3333 nM T68251 CTB9P6 44440461 Ki = 307 nM T68251 C63RLK 44440462 Ki > 3333 nM T68251 C23JBO 44440463 Ki > 3333 nM T68251 CT9P3Y 44440464 Ki > 3333 nM T68251 CX32AM 44440465 Ki > 3333 nM T68251 C6FOC7 44440466 Ki > 3333 nM T68251 CMPX37 44440467 Ki > 3333 nM T68251 CV4F6Z 44440468 Ki > 3333 nM T68251 C6K8VB 44440469 Ki > 3333 nM T68251 C4Y0UM 44440470 Ki > 3333 nM T68251 CHU49A 44440471 Ki > 3333 nM T68251 C8OI4L 44440472 Ki > 3333 nM T68251 CV58YW 44441018 Ki > 3333 nM T68251 CV85PN 44441019 Ki > 3333 nM T68251 C5O2WK 44441020 Ki > 3333 nM T68251 CU67WS 44441021 Ki > 3333 nM T68251 CXZ53B 44441022 Ki > 3333 nM T68251 C8S7UT 44441023 Ki > 3333 nM T68251 CT4PZ9 44441024 Ki > 3333 nM T68251 CU9GE6 44441025 Ki > 3333 nM T68251 CB2IT4 44441026 Ki > 3333 nM T68251 CN4X2F 44441027 Ki > 3333 nM T68251 CPF45Y 44441028 Ki > 3333 nM T68251 CAM23N 44441029 Ki > 3333 nM T68251 C23BPG 44441030 Ki > 3333 nM T68251 C5YMT6 44441031 Ki > 3333 nM T68251 C9A6GJ 44441032 Ki > 3333 nM T68251 CYSU19 44441033 Ki > 3333 nM T68251 CB9P0C 44442303 IC50 = 870 nM T68251 C7HO0Y 44442304 IC50 = 1630 nM T68251 CAR3S2 44442305 IC50 = 960 nM T68251 CZK0A9 44442306 IC50 = 2230 nM T68251 C71MCV 44442307 IC50 = 840 nM T68251 CN70HO 44442308 IC50 = 520 nM T68251 CVE5P0 44442309 IC50 = 1110 nM T68251 C3PT7N 44442310 IC50 = 840 nM T68251 CGS18B 44442311 IC50 = 1620 nM T68251 CIZL27 44442312 IC50 = 760 nM T68251 CCFV76 44442313 IC50 = 700 nM T68251 C4HYM6 44442314 IC50 = 260 nM T68251 CZ2PE6 44442315 IC50 = 1030 nM T68251 C3I7RG 44442317 IC50 = 2570 nM T68251 CGR6E7 44442318 IC50 = 1230 nM T68251 C97ZHM 44442319 IC50 = 1450 nM T68251 C3DIB8 44442320 IC50 = 1000 nM T68251 C0HX1L 44445199 IC50 = 67000 nM T68251 CPQT35 44445200 IC50 = 66000 nM T68251 C2X6IP 44445201 IC50 = 72000 nM T68251 CSRB79 44445202 IC50 = 70000 nM T68251 C2O6KZ 44445203 IC50 = 101000 nM T68251 CASF34 44445204 IC50 = 65000 nM T68251 CQZ6M0 44445205 IC50 = 69000 nM T68251 CH7Z5M 44445206 IC50 = 73000 nM T68251 C71CPO 44445207 IC50 > 150 nM T68251 CO9QA4 44445209 IC50 = 70000 nM T68251 CH3UQ5 44445210 IC50 = 110000 nM T68251 C6B4LG 44445211 IC50 > 150 nM T68251 C1WA5N 44445212 IC50 = 90000 nM T68251 CM2CD0 44445213 IC50 = 71000 nM T68251 C6ZX2P 44445214 IC50 = 70000 nM T68251 C9KE8P 44445215 IC50 = 71000 nM T68251 C68QEF 44445216 IC50 = 66000 nM T68251 CCK7W2 44445217 IC50 = 70000 nM T68251 C58BQA 44445218 IC50 = 69000 nM T68251 C4CGN2 44445219 IC50 = 39000 nM T68251 C1IVR6 44445220 IC50 = 86000 nM T68251 CG2U7H 44445221 IC50 = 64000 nM T68251 CVW48J 44445222 IC50 = 69000 nM T68251 CL3HZ8 44445223 IC50 = 69000 nM T68251 CPY73U 44445224 IC50 = 57000 nM T68251 C9MA2F 44445225 IC50 = 68000 nM T68251 C9SJM3 44445226 IC50 = 107000 nM T68251 CH91WG 44445228 IC50 = 90000 nM T68251 CO59HI 44445229 IC50 = 109000 nM T68251 C62WPE 44445230 IC50 = 125000 nM T68251 COIR35 44445231 IC50 = 107000 nM T68251 CBH0M7 44445233 IC50 = 33000 nM T68251 CIS7M5 44445234 IC50 > 150 nM T68251 CKN60A 44445235 IC50 = 73000 nM T68251 CP4XL8 44445237 IC50 = 65000 nM T68251 CJA79R 44445239 IC50 = 111000 nM T68251 CA72BI 44445240 IC50 = 103000 nM T68251 CZJB48 44445241 IC50 > 150000 nM T68251 C85EVH 44445242 IC50 > 150000 nM T68251 C9DI7F 44445243 IC50 = 73000 nM T68251 CVLH67 44445244 IC50 = 85000 nM T68251 CIP3X8 44445245 IC50 = 119000 nM T68251 CL1MK6 44445246 IC50 = 100000 nM T68251 C0CX7T 44445247 IC50 = 7000 nM T68251 CEZ2P7 44445248 IC50 = 98000 nM T68251 CL0K9Q 44445249 IC50 = 110000 nM T68251 C9T2SH 44445250 IC50 = 125000 nM T68251 C5EFP9 44445251 IC50 = 90000 nM T68251 CLJ71G 44445252 IC50 = 91000 nM T68251 C8TF3E 44445253 IC50 = 63000 nM T68251 C4CAY7 44445254 IC50 = 124000 nM T68251 CH1LE5 44445255 IC50 = 108000 nM T68251 CLP96W 44445256 IC50 = 66000 nM T68251 CK8S4Z 44445257 IC50 = 79000 nM T68251 C03EJW 44445258 IC50 = 90000 nM T68251 CO9SM5 44445261 IC50 = 96000 nM T68251 C3FX8B 44445262 IC50 = 108000 nM T68251 CZS8N5 44445263 IC50 = 98000 nM T68251 CMW2U6 44445264 IC50 = 100000 nM T68251 CB47AH 44445265 IC50 = 110000 nM T68251 CA43LS 44445266 IC50 = 42000 nM T68251 C23MDF 44445267 IC50 = 46000 nM T68251 C9K3DI 44445268 IC50 = 93000 nM T68251 C2ZAK4 44445269 IC50 = 77000 nM T68251 CIVC64 44445270 IC50 = 85000 nM T68251 C8W1HX 44445271 IC50 > 150000 nM T68251 CTFR27 44445272 IC50 > 150000 nM T68251 C20DNO 44445273 IC50 > 150000 nM T68251 CWLC15 44445274 IC50 > 150000 nM T68251 CZD5M3 44445275 IC50 > 150000 nM T68251 CJET46 44445276 IC50 > 150000 nM T68251 CI58AM 44445277 IC50 = 149000 nM T68251 CDN37V 44445278 IC50 > 150000 nM T68251 CE36AB 44445279 IC50 > 150000 nM T68251 CV9KX5 44445280 IC50 > 150000 nM T68251 C4S2WX 44445281 IC50 > 150000 nM T68251 C0HXS4 44445391 IC50 = 620 nM T68251 CT1CP7 44445392 IC50 = 4380 nM T68251 CRNK10 44445393 IC50 = 3080 nM T68251 CF0LR3 44445394 IC50 = 776 nM T68251 C9WQ8E 44445790 IC50 = 3.388 nM T68251 CEGL68 44445796 IC50 = 3981.07 nM T68251 CH2Y7W 44445813 Ki = 2.1 nM T68251 C4J2QM 44445814 Ki = 6.1 nM T68251 CP5H1Q 44446267 IC50 = 6 nM T68251 C30TQK 44446273 IC50 = 1470 nM T68251 CB76CO 44446275 IC50 = 860 nM T68251 C20HIJ 44446753 IC50 = 13 nM T68251 C9CS8E 44446754 IC50 = 21 nM T68251 C4Z7IQ 44446755 IC50 = 50 nM T68251 C4K5QT 44446756 IC50 = 1100 nM T68251 CZEH45 44446757 IC50 = 24 nM T68251 C47SRV 44446758 IC50 = 433 nM T68251 C8CVO1 44446759 IC50 = 2500 nM T68251 C8HM5N 44446763 IC50 = 159 nM T68251 CU5Z4V 44446765 IC50 = 14 nM T68251 C9USL8 44446766 IC50 = 4999 nM T68251 CYO65B 44446797 IC50 = 63 nM T68251 CPI3T0 44446799 IC50 < 5 nM T68251 CGH0A2 44446805 IC50 = 32 nM T68251 CH72RW 44446806 IC50 > 5000 nM T68251 CTKX08 44446807 IC50 = 391 nM T68251 CJ1MP7 44446808 IC50 = 1387 nM T68251 CJN1L7 44446821 IC50 = 39 nM T68251 C4LF6Y 44446822 Ki = 302 nM T68251 C9FG5A 44446823 IC50 = 35 nM T68251 C1P0BV 44446824 IC50 = 37 nM T68251 C5AW3N 44446825 IC50 = 50 nM T68251 C17YSI 44446827 IC50 = 53 nM T68251 C3O8AX 44446835 IC50 = 472 nM T68251 CE2OM1 44446839 IC50 = 106 nM T68251 C49VJF 44446842 IC50 = 86 nM T68251 CF4DL2 44446843 IC50 = 960 nM T68251 C8OS4K 44446845 IC50 > 5000 nM T68251 CIP23G 44447330 IC50 = 10 nM T68251 CPS5M4 44447343 IC50 = 64 nM T68251 CB3F0E 44447344 IC50 = 53 nM T68251 C6WSC7 44447346 IC50 = 52 nM T68251 C6MOB0 44447348 IC50 = 549 nM T68251 CM7JV0 44447353 IC50 = 13 nM T68251 CY2XR5 44447363 IC50 = 1400 nM T68251 CU2BC6 44447364 IC50 > 10000 nM T68251 CXS34M 44447371 IC50 = 262 nM T68251 CD8RX4 44447437 IC50 > 2000 nM T68251 CLNK98 44447442 IC50 > 2000 nM T68251 CA5J9Q 44454525 IC50 > 10000 nM T68251 C6L1OH 44454554 IC50 = 283 nM T68251 CHTY64 44454555 IC50 = 297 nM T68251 CLNM62 44454612 IC50 = 247 nM T68251 CZ2QY4 44454641 IC50 = 344 nM T68251 C7DIB0 44454661 IC50 = 401 nM T68251 CTR91D 44454664 IC50 = 582 nM T68251 CR3PO9 44454741 IC50 = 1262 nM T68251 C1ZSK0 44454742 IC50 = 286 nM T68251 CM8AG1 44454790 IC50 = 2917 nM T68251 CCH42M 44454856 IC50 = 893 nM T68251 CQG09B 44454861 IC50 = 61 nM T68251 CQ5YK3 44454864 IC50 = 73 nM T68251 CLG57Z 44454888 IC50 = 2317 nM T68251 CMEJ96 44454891 IC50 = 147 nM T68251 CV07DO 44455123 IC50 = 4591 nM T68251 C9MHD2 44455124 IC50 = 108.4 nM T68251 C2L1VK 44455161 IC50 = 5.7 nM T68251 C4CZ7N 44455196 IC50 = 4.9 nM T68251 CZ15QG 44455197 IC50 = 104.5 nM T68251 CJ6L1K 44455200 IC50 = 1.7 nM T68251 CLK5O7 44455240 IC50 = 6.1 nM T68251 CSKN69 44455242 IC50 = 5 nM T68251 C3U9VM 44455265 IC50 = 22.4 nM T68251 CG65TZ 44455266 IC50 = 6.5 nM T68251 C14QTI 44455267 IC50 = 41 nM T68251 CSX4F2 44455294 IC50 = 6.1 nM T68251 CJ29BT 44455298 IC50 = 66.4 nM T68251 CCK15P 44455331 IC50 = 66.2 nM T68251 CW8IB7 44455332 IC50 = 662 nM T68251 C9ZXF4 44455360 IC50 = 242 nM T68251 CFB78A 44455363 IC50 > 1000 nM T68251 CW46RV 44455498 Ki = 1500 nM T68251 CXNP45 44455499 Ki = 2733 nM T68251 C6CED5 44455528 Ki > 3333 nM T68251 CUQH30 44455553 Ki = 1700 nM T68251 C83KYJ 44455582 Ki > 3333 nM T68251 CK5N1S 44455612 Ki > 3333 nM T68251 CU2E7V 44455613 Ki > 3333 nM T68251 CH1DI4 44455614 Ki > 3333 nM T68251 CFQ79A 44455647 Ki > 3333 nM T68251 C3J1SV 44455676 IC50 = 36.8 nM T68251 CS6HL1 44455704 IC50 > 1000 nM T68251 CR4EX3 44455706 IC50 > 1000 nM T68251 CC01WS 44455737 IC50 = 377 nM T68251 C0R9SH 44455760 IC50 = 167.5 nM T68251 C6FV2Z 44455783 Ki > 3333 nM T68251 C7W6XV 44455786 IC50 = 72 nM T68251 CO58GJ 44455787 IC50 = 184 nM T68251 CPYV60 44455807 Ki = 2633 nM T68251 CLAT19 44455811 IC50 > 1000 nM T68251 C3TS1X 44455813 IC50 = 10.6 nM T68251 C92AFN 44455816 IC50 = 84.5 nM T68251 CGA0T4 44455829 Ki > 3333 nM T68251 CIR06N 44455835 IC50 = 16.7 nM T68251 C38VBL 44455836 IC50 = 17.2 nM T68251 CKB6E7 44455837 IC50 = 468 nM T68251 CV2B4N 44455858 Ki > 3333 nM T68251 CL6UY9 44455865 IC50 > 1000 nM T68251 CVR58Q 44455879 Ki > 3333 nM T68251 CWZ8K6 44455880 Ki > 3333 nM T68251 CEN93Y 44460382 Ki > 10000 nM T68251 CL30OP 44460588 Ki = 220 nM T68251 C0A1KH 44460605 Ki = 77 nM T68251 CDN1V6 44460606 Ki = 110 nM T68251 CJ6PN3 44460646 Ki = 11 nM T68251 CU8A1O 44460672 Ki = 6100 nM T68251 CIQ87B 44460676 Ki = 4840 nM T68251 C5B8NZ 44460690 Ki = 12 nM T68251 CK4WU2 44460737 Ki = 130 nM T68251 CG0Z7I 44478924 IC50 = 1300 nM T68251 CFO27Y 44478926 IC50 = 230 nM T68251 CBZJ29 44478927 IC50 = 9.7 nM T68251 CRJ24K 44479197 IC50 = 7 nM T68251 CGOH82 44479198 IC50 = 710 nM T68251 CLV56M 44479199 IC50 = 47 nM T68251 CY92OQ 44479458 IC50 = 9900 nM T68251 CH1QG9 44479459 IC50 = 100 nM T68251 CB1NT7 44479460 IC50 = 38 nM T68251 C0JQ9L 44479699 IC50 = 73 nM T68251 C0DN1Q 44479700 IC50 = 58000 nM T68251 CTG24W 44479702 IC50 = 2400 nM T68251 CGZ49M 44479703 IC50 = 190 nM T68251 CAK94X 44563337 IC50 = 193 nM T68251 CSH4K3 44563364 IC50 = 10000 nM T68251 CAF95R 44563365 IC50 = 10000 nM T68251 CO4FQ1 44563366 IC50 = 10000 nM T68251 C6WA3X 44563401 IC50 = 10000 nM T68251 CX5L7N 44563402 IC50 = 24 nM T68251 CJ8V4U 44563403 IC50 = 18 nM T68251 CN2BM4 44563404 IC50 = 100 nM T68251 C3KCV6 44563405 IC50 = 740 nM T68251 CI0R5M 44563465 IC50 = 310 nM T68251 C5IQ9Z 44563466 IC50 = 320 nM T68251 C6ZEW9 44563467 IC50 = 1400 nM T68251 CZ2EL1 44563468 IC50 = 300 nM T68251 CDV6R7 44563469 IC50 = 92 nM T68251 CJ2BU5 44563487 IC50 = 37 nM T68251 CP54WT 44563489 IC50 = 1813 nM T68251 C1UXP6 44563490 IC50 = 310 nM T68251 CZ0W1A 44563491 IC50 = 1273 nM T68251 C37UAM 44563492 IC50 = 65 nM T68251 C4BD0N 44563493 IC50 = 247 nM T68251 CNP6M7 44563494 IC50 = 45 nM T68251 C0J6LB 44563970 IC50 = 2600 nM T68251 CR6NO2 44564180 IC50 = 6 nM T68251 C3US0I 44569010 IC50 = 3200 nM T68251 C3TAN1 44569011 IC50 = 2200 nM T68251 CF0L2W 44569012 IC50 = 50 nM T68251 CGI35S 44569013 IC50 = 200 nM T68251 C8PO5Q 44569024 IC50 = 40 nM T68251 C52JXP 44569036 IC50 = 3500 nM T68251 CU1NI6 44569037 IC50 = 2700 nM T68251 CS9CH4 44569038 IC50 = 40 nM T68251 C63ZQK 44569039 IC50 = 10 nM T68251 C2WE7H 44569040 IC50 = 1300 nM T68251 CO8FB4 44569058 IC50 = 90 nM T68251 C3K4ED 44569059 IC50 = 5200 nM T68251 CPWR76 44569060 IC50 = 1500 nM T68251 CU39FK 44569061 IC50 = 200 nM T68251 CR6H0X 44569062 IC50 = 700 nM T68251 CTWR37 44569063 IC50 = 8900 nM T68251 C6M9SH 44569081 IC50 = 500 nM T68251 C5RN7U 44569082 IC50 = 4 nM T68251 CQ9OA7 44569083 IC50 = 20 nM T68251 C70UVG 44571513 IC50 = 50500 nM T68251 CCV74H 44576563 IC50 = 400 nM T68251 C59TCG 44576564 IC50 = 2000 nM T68251 CMI9S4 44576565 IC50 = 9500 nM T68251 CD8ZI4 44576587 IC50 = 100 nM T68251 CQ87CS 44576614 IC50 = 200 nM T68251 CJY2W3 44576615 IC50 = 300 nM T68251 CL92CH 44576616 IC50 = 200 nM T68251 CIU84E 44576617 IC50 = 1100 nM T68251 C9ODS1 44576618 IC50 = 1500 nM T68251 C35DWL 44576631 IC50 = 6 nM T68251 C6ZL1U 44576632 IC50 = 8 nM T68251 CK09LV 44576633 IC50 = 8 nM T68251 CFL76T 44576634 IC50 = 11 nM T68251 CC58GQ 44576635 IC50 = 12 nM T68251 CPT42K 44580109 IC50 > 5000 nM T68251 CQ7W5I 44580110 Ki > 3000 nM T68251 CWD32S 44580184 IC50 = 664 nM T68251 CQ4ZR1 44580422 IC50 = 750 nM T68251 C0XJ5C 44580496 Ki > 3333 nM T68251 CK68GT 44580539 Ki = 1.37 nM T68251 CXIY57 44580801 Ki > 10000000 nM T68251 C0OA8Y 44580802 Ki > 10000000 nM T68251 CNC4D7 44581071 Ki = 7000000 nM T68251 CDF48U 44581111 Ki > 10000000 nM T68251 C06BRD 44582547 IC50 = 107200 nM T68251 C51VNE 44582548 IC50 = 287300 nM T68251 CLK3R4 44582549 IC50 = 76800 nM T68251 CZTW24 44582550 IC50 = 52800 nM T68251 CP0AJ7 44582568 IC50 = 59900 nM T68251 CCZ07T 44582586 IC50 = 76100 nM T68251 CN58BM 44582588 IC50 = 71200 nM T68251 C3UJ2Q 44582621 IC50 = 659600 nM T68251 C35BEJ 44582622 IC50 = 501500 nM T68251 C3UE5R 44582644 IC50 = 116300 nM T68251 CX1GV0 44582645 IC50 = 71400 nM T68251 C3IU2S 44582646 IC50 = 64300 nM T68251 C63ODU 44582647 IC50 = 120800 nM T68251 C7EAZ1 44582685 IC50 = 235800 nM T68251 CZW4O6 44582686 IC50 = 159100 nM T68251 C3AX6W 44582687 IC50 = 211400 nM T68251 CC0LO7 44582688 IC50 = 283600 nM T68251 CX63IA 44582689 IC50 = 256100 nM T68251 CL73BH 44582717 IC50 = 79600 nM T68251 CY2PM8 44582718 IC50 = 83200 nM T68251 C9EPQ6 44582719 IC50 = 76800 nM T68251 CF1G7I 44582720 IC50 = 101500 nM T68251 C15RUQ 44582746 IC50 = 76500 nM T68251 C3CJD0 44582747 IC50 = 397600 nM T68251 C16RAH 44582748 IC50 = 368100 nM T68251 CQ9XG5 44582769 IC50 = 470600 nM T68251 C7UTR1 44582771 IC50 = 470700 nM T68251 CE2D6Z 44582793 IC50 = 340800 nM T68251 CUR8M1 44582868 IC50 = 55300 nM T68251 CNK9C7 44582869 IC50 = 628000 nM T68251 CX49HN 44582873 IC50 = 369400 nM T68251 C56WPA 44582874 IC50 = 169400 nM T68251 C8TGB1 44582875 IC50 = 114900 nM T68251 CYV0N5 44582876 IC50 = 26100 nM T68251 CR4SF2 44582887 IC50 = 52300 nM T68251 C50OTD 44582888 IC50 = 54400 nM T68251 CDX63O 44582890 IC50 = 33600 nM T68251 C6X0FM 44582904 IC50 = 71200 nM T68251 CY3N7I 44582905 IC50 = 86300 nM T68251 CY4A6F 44582906 IC50 = 108700 nM T68251 CD0J5R 44582907 IC50 = 122400 nM T68251 C2Z4HB 44583600 IC50 = 1277 nM T68251 CD4Q8C 44583601 IC50 = 8 nM T68251 CD2AQ7 44583620 IC50 = 92 nM T68251 CLZ6X5 44583621 IC50 = 81 nM T68251 C5HA4P 44583622 IC50 = 180 nM T68251 C7PR8I 44583623 IC50 = 106 nM T68251 CDRC42 44583654 IC50 = 100 nM T68251 C5HEX6 44583655 IC50 = 1090 nM T68251 CM79HD 44583656 IC50 > 5000 nM T68251 C20FCM 44583672 IC50 > 5000 nM T68251 CLAU98 44586492 IC50 = 8760 nM T68251 CY8X7P 44586493 IC50 = 2930 nM T68251 CDS86C 44586529 IC50 = 3140 nM T68251 COD20L 44586530 IC50 = 12700 nM T68251 C1W2SV 44586531 IC50 = 17800 nM T68251 C5S0OJ 44586532 IC50 = 50500 nM T68251 CB2P7I 44586533 IC50 = 7480 nM T68251 CKRT49 44586578 IC50 = 19200 nM T68251 C8XY1Z 44586579 IC50 = 13100 nM T68251 CE9BZ5 44586580 IC50 = 25500 nM T68251 CXDF71 44586581 IC50 = 14300 nM T68251 COFY06 44586582 IC50 = 8080 nM T68251 CI2PT3 44586626 IC50 = 8000 nM T68251 C4GQ6Y 44586627 IC50 = 12600 nM T68251 CTO94B 44586628 IC50 = 3540 nM T68251 C9Y0CR 44586662 IC50 = 11700 nM T68251 CBV5P8 44586663 IC50 = 32000 nM T68251 C2U0CY 44586664 IC50 = 9940 nM T68251 C1IBA2 44588219 IC50 = 151400 nM T68251 C6XE5V 44588251 IC50 = 771900 nM T68251 C1UW6M 44588252 IC50 = 802300 nM T68251 CXF40R 44588253 IC50 = 78800 nM T68251 CQF2I5 44588254 IC50 = 546800 nM T68251 CBA1Y8 44588279 IC50 > 1000000 nM T68251 C8RI4Q 44591819 IC50 = 30000 nM T68251 C6BXS2 44591880 IC50 = 37700 nM T68251 CM9IN6 44592481 IC50 = 14400 nM T68251 CZNQ90 44593458 IC50 = 9 nM T68251 CR3Q4N 44593532 IC50 = 7100 nM T68251 CH8QS0 44596287 IC50 = 128 nM T68251 CTW7F2 44601281 IC50 = 1.6 nM T68251 CW5A2D 44608129 IC50 = 86 nM T68251 CT7KX5 44608938 IC50 = 96 nM T68251 CJRP30 44608939 IC50 = 458 nM T68251 COI5K3 44608942 IC50 = 706 nM T68251 CS4C5T 44609098 IC50 = 200 nM T68251 CMLV87 44609099 IC50 = 706 nM T68251 C3T9SV 44609100 IC50 = 54 nM T68251 C19LWR 44634267 IC50 = 0.13 nM T68251 CM0I4J 45101511 IC50 = 1475 nM T68251 CZP79X 45268488 IC50 = 379 nM T68251 CK50JB 45268522 IC50 = 8990 nM T68251 C2B0GI 45268787 Ki = 1 nM T68251 CVG5I2 45269378 IC50 = 4000 nM T68251 CQC5Y4 45269386 IC50 = 2840 nM T68251 CACH13 45269631 IC50 = 12 nM T68251 CTOH60 45270200 IC50 = 4410 nM T68251 C2H5IY 45271017 IC50 = 3590 nM T68251 C0YT8W 45271893 IC50 = 1150 nM T68251 CVNO86 45271894 IC50 = 1410 nM T68251 C7OQB3 45271912 IC50 = 2470 nM T68251 C3SWC7 45272759 IC50 = 7500 nM T68251 CH4NL1 45376336 IC50 = 1937.23 nM T68251 C36HRP 45377138 IC50 > 22000 nM T68251 C6B7ZY 45377564 IC50 > 500000 nM T68251 C5HAR6 45377565 IC50 > 20000 nM T68251 CKR0Q8 45377703 IC50 > 24000 nM T68251 C3SQL2 45378250 IC50 = 190 nM T68251 CQE49A 45378251 IC50 = 1.5 nM T68251 CO4AC6 45378252 IC50 = 17 nM T68251 C42FPG 45378253 IC50 = 4.2 nM T68251 CI82BN 45378254 IC50 = 21 nM T68251 C6MY2W 45380188 IC50 = 190 nM T68251 C9P0DG 45380189 IC50 = 29 nM T68251 CRY0E8 45380190 IC50 = 0.7 nM T68251 C0MPH3 45380191 IC50 = 390 nM T68251 CMPE63 45482676 IC50 = 1500 nM T68251 CZS39O 45487302 IC50 = 210 nM T68251 C4ZWY7 45487310 IC50 = 432 nM T68251 C9SV0H 45487311 IC50 = 581 nM T68251 C6GCM7 45487332 IC50 < 5 nM T68251 CCF05Q 45487333 IC50 = 102 nM T68251 C23NRD 45487334 IC50 > 2000 nM T68251 CY09ZU 45487335 IC50 = 344 nM T68251 CQHJ85 45487342 IC50 = 11 nM T68251 C3ZLN1 45487343 IC50 = 12 nM T68251 CI6DW2 45487357 IC50 < 5 nM T68251 COX40Y 45487358 IC50 = 102 nM T68251 CF1T7M 45487359 IC50 = 843 nM T68251 CRXI29 45487373 IC50 > 2000 nM T68251 CYL32E 45487376 IC50 = 235 nM T68251 CO5P9I 45487386 IC50 = 506 nM T68251 CS9Y8G 45487387 IC50 > 2000 nM T68251 CAN4J2 45487388 IC50 = 1662 nM T68251 CWLC18 45487393 IC50 = 471 nM T68251 CO9NJ2 45487398 IC50 = 365 nM T68251 CDN5Q6 45487399 IC50 = 502 nM T68251 CI4KJ5 45487400 IC50 = 613 nM T68251 C49HOI 45487401 IC50 = 730 nM T68251 CBK43U 45487402 IC50 < 5 nM T68251 C56WVI 46184724 Ki > 50000 nM T68251 CMB53L 46212112 IC50 = 159390 nM T68251 CX58KQ 46212114 IC50 = 58220 nM T68251 C9PXD0 46212116 IC50 = 17170 nM T68251 C6KHO2 46212117 IC50 = 36040 nM T68251 C9XGD0 46212861 IC50 = 187410 nM T68251 CLWA85 46228171 IC50 > 1000000 nM T68251 CFQ67J 46228182 IC50 > 1000000 nM T68251 CCV7T2 46228183 IC50 > 1000000 nM T68251 CU2WI8 46228191 IC50 > 1000000 nM T68251 CT6JZ9 46228192 IC50 = 594300 nM T68251 C6H7AB 46228205 IC50 = 999000 nM T68251 CJ9SD0 46228215 IC50 = 447200 nM T68251 C7WS9P 46228222 IC50 > 1000000 nM T68251 C71RSJ 46228223 IC50 > 1000000 nM T68251 CKCE97 46228233 IC50 > 1000000 nM T68251 CWUG47 46228234 IC50 = 324400 nM T68251 CM3YZ1 46228235 IC50 > 1000000 nM T68251 CYUM78 46228241 IC50 > 1000000 nM T68251 C6HCD2 46228242 IC50 > 1000000 nM T68251 C0GX8M 46228245 IC50 > 1000000 nM T68251 C9FM5N 46228246 IC50 = 176500 nM T68251 C4KA1Y 46228247 IC50 > 1000000 nM T68251 C7HIE4 46228248 IC50 = 131000 nM T68251 CQVZ58 46228249 IC50 > 1000000 nM T68251 C5WV8N 46228250 IC50 > 1000000 nM T68251 CR0BP8 46228264 IC50 > 1000000 nM T68251 CGW3Q4 46228265 IC50 > 1000000 nM T68251 CVN7J0 46228266 IC50 = 166600 nM T68251 C51LDC 46228283 IC50 > 1000000 nM T68251 C2JVF4 46228308 IC50 = 196600 nM T68251 C7Z6XB 46228317 IC50 > 1000000 nM T68251 C0S8FV 46231953 IC50 = 400 nM T68251 CN3OS2 46232362 IC50 = 6460800 nM T68251 CF9D2G 46232363 IC50 = 124320 nM T68251 C5GT8X 46232364 IC50 = 624480 nM T68251 C9A8BO 46232365 IC50 = 2000000 nM T68251 CP49KE 46232415 IC50 = 24180 nM T68251 CFZX82 46232416 IC50 = 26170 nM T68251 C3L7VK 46232417 IC50 = 1362800 nM T68251 C4XOU1 46232418 IC50 = 56600 nM T68251 C1S8BQ 46232490 IC50 = 106000 nM T68251 CAV06U 46232491 IC50 = 105300 nM T68251 CVF9D5 46232492 IC50 = 9426500 nM T68251 C18JTQ 46232493 IC50 = 1750000 nM T68251 CFA58J 46232533 IC50 = 2757800 nM T68251 C9C7IE 46232534 IC50 = 11520000 nM T68251 CFU05P 46232535 IC50 = 1920500 nM T68251 CSU81E 46233057 IC50 = 58140 nM T68251 C8SM5H 46233058 IC50 = 30050 nM T68251 C8W7RP 46233059 IC50 = 10490 nM T68251 C3IA9P 46233060 IC50 = 37290 nM T68251 CZ6C8P 46703060 IC50 = 5.97 nM T68251 C0DHL4 46703061 IC50 = 1721.82 nM T68251 CYA45K 46703062 IC50 = 3.55 nM T68251 CY72WL 46703063 IC50 = 5.27 nM T68251 C1YHS2 46703064 IC50 = 1679.56 nM T68251 C8HX7K 46840956 IC50 = 45820 nM T68251 CH0Z1E 46844314 Ki = 1208 nM T68251 C8MR0H 46847340 IC50 = 4000 nM T68251 C20BTY 46856241 Ki = 43600 nM T68251 C0ECU2 46861775 IC50 = 8.95 nM T68251 C0Y9NZ 46861793 IC50 = 8.31 nM T68251 C2S4YC 46866644 IC50 = 15000 nM T68251 C7QR8Y 46866645 IC50 = 10000 nM T68251 CUH07J 46866646 IC50 = 7000 nM T68251 C8GK4C 46866647 IC50 = 4000 nM T68251 C5L8GF 46871738 IC50 = 12.1 nM T68251 CR1KF7 46871739 IC50 = 3.7 nM T68251 C8Q6YR 46871740 IC50 = 5.3 nM T68251 C58YSM 46871741 IC50 = 6000 nM T68251 C3X5EN 46873064 IC50 = 53670 nM T68251 CR96AK 46890762 IC50 > 10000 nM T68251 C5G9FX 46890763 IC50 = 1400 nM T68251 COP78K 46890764 IC50 = 4500 nM T68251 C60QSB 46890765 IC50 = 1600 nM T68251 CQ5P9V 46890766 IC50 = 700 nM T68251 CB90YN 46890767 IC50 = 5600 nM T68251 CUA7L6 46890821 IC50 = 3600 nM T68251 C9BNQ7 46890822 IC50 = 1600 nM T68251 CTF20Y 46890823 IC50 = 1750 nM T68251 CR3QW7 46891107 IC50 = 21.1 nM T68251 C5MK3A 46891108 IC50 = 88 nM T68251 CQ5E1H 46891109 IC50 = 40 nM T68251 C0NW9D 46891110 IC50 = 370 nM T68251 C91LGI 46891170 IC50 = 48.5 nM T68251 CGI5B4 46891171 IC50 = 330 nM T68251 CZPM12 46891172 IC50 = 18.4 nM T68251 C2V6MW 46891173 IC50 = 35 nM T68251 CZWT45 46891207 IC50 = 1400 nM T68251 CFE58Q 46891208 IC50 = 5.4 nM T68251 C8S7QX 46891209 IC50 = 32.6 nM T68251 C5Y0MN 46891255 IC50 = 3700 nM T68251 CJ16SE 46891256 IC50 = 2 nM T68251 C7Y9TE 46891257 IC50 = 82 nM T68251 C7DT6W 46891258 IC50 = 700 nM T68251 CLF7Y4 46891311 IC50 = 900 nM T68251 C2IN7Y 46891312 IC50 = 3100 nM T68251 CNXU57 46891313 IC50 = 70 nM T68251 CJB5D0 46891314 IC50 = 5400 nM T68251 CVK0E5 46891356 IC50 = 500 nM T68251 C89RPO 46891357 IC50 = 505 nM T68251 CVB6K4 46891358 IC50 = 1750 nM T68251 C67WEK 46891359 IC50 = 800 nM T68251 CPQ37V 46891414 IC50 > 10000 nM T68251 C5LTI6 46891459 IC50 = 2900 nM T68251 C92FBL 46891460 IC50 = 2100 nM T68251 C1A0OE 46891522 IC50 = 2100 nM T68251 C2I6FV 46891523 IC50 = 2400 nM T68251 CAZ9Q5 46891524 IC50 = 7300 nM T68251 CG02KB 46891525 IC50 = 1700 nM T68251 C7ZG8J 46891526 IC50 > 10000 nM T68251 CRQ13J 46891580 IC50 = 2500 nM T68251 CERM39 46891581 IC50 = 5500 nM T68251 CN8WF9 46891582 IC50 = 7000 nM T68251 C86RLM 46891583 IC50 = 900 nM T68251 CM7S5T 46891584 IC50 = 6000 nM T68251 CRY18A 46891617 IC50 = 900 nM T68251 C0F7SU 46905989 IC50 = 112000 nM T68251 C49PYF 46907509 IC50 = 8.92 nM T68251 C2U1GW 46907510 IC50 = 9.11 nM T68251 C7MUS8 46907512 IC50 = 1820.53 nM T68251 C71YRF 46907513 IC50 = 1873.02 nM T68251 CVH58U 46907580 IC50 = 8.3 nM T68251 C0S9WB 46919610 Ki = 1900 nM T68251 CXDL74 46927871 IC50 = 8270 nM T68251 CE3H7I 46938726 IC50 < 0.1 nM T68251 C9T0HR 46938727 IC50 < 0.1 nM T68251 C0YR7M 46938728 IC50 < 0.1 nM T68251 C2TE8J 47162079 IC50 = 60000 nM T68251 CC42DK 49863560 IC50 = 129000 nM T68251 C4UWB6 49863561 IC50 = 18500 nM T68251 CMR3B0 49863562 IC50 = 121000 nM T68251 CBE6H5 49863563 IC50 = 127000 nM T68251 CR0I9V 49863564 IC50 = 12000 nM T68251 CD17YP 49863589 IC50 = 272000 nM T68251 CXW4C6 49863590 IC50 = 107000 nM T68251 C1B6ZU 49863591 IC50 = 155000 nM T68251 C0S2OT 49863592 IC50 > 1000000 nM T68251 CT3W2H 49863593 IC50 > 1000000 nM T68251 CG96WY 49863619 IC50 = 22700 nM T68251 CG40UX 49863620 IC50 = 315650 nM T68251 C0IX5P 49863621 IC50 > 1000000 nM T68251 CSC7K2 49863622 IC50 = 141000 nM T68251 C1FLD5 49863915 IC50 = 122000 nM T68251 CL90XE 49863932 IC50 > 1000000 nM T68251 CXZ8Y3 49863933 IC50 = 60400 nM T68251 CKXZ37 49863934 IC50 = 62700 nM T68251 CFD6O0 49863953 IC50 = 71600 nM T68251 C1L6TV 49863954 IC50 = 131000 nM T68251 CEL71O 49863955 IC50 = 46900 nM T68251 CJB0T7 49863956 IC50 = 454000 nM T68251 C7S9QA 50913428 IC50 > 500000 nM T68251 CO4XE9 50913573 IC50 > 500000 nM T68251 C2T1AZ 50925490 IC50 = 3000 nM T68251 CJG7H2 50941564 IC50 = 8800 nM T68251 C5B6SP 50941565 IC50 = 7200 nM T68251 CV4BM3 50941566 IC50 = 10800 nM T68251 C29WVD 50941567 IC50 = 8400 nM T68251 CKN8Z0 50941568 IC50 = 5600 nM T68251 CQ64FL 50941569 IC50 = 3900 nM T68251 CC4V0N 50941747 IC50 = 4300 nM T68251 C7AU4S 50943150 IC50 > 100000 nM T68251 CXF4V3 50990921 IC50 > 6300 nM T68251 CAS94N 51346773 Ki = 390 nM T68251 CP65WT 51346774 Ki = 90 nM T68251 C5OIA2 51346775 Ki = 280 nM T68251 CU2SX3 51355576 Ki > 10000 nM T68251 CQM4E7 52936345 IC50 = 19 ug.mL-1 T68251 CLA96C 53232689 Ki = 400 nM T68251 C3BGW0 53233015 Ki = 20500 nM T68251 CZ06OY 53233469 IC50 = 360 nM T68251 CMQZ70 53242178 IC50 > 23000 nM T68251 CC9HK5 53245646 IC50 = 6309.57 nM T68251 CRI92N 53311230 IC50 > 10000 nM T68251 C74CKF 53318123 Ki = 61 nM T68251 C47DIU 53318911 IC50 = 120 nM T68251 CC6DR2 53318912 IC50 = 4200 nM T68251 C7V1NC 53320225 IC50 = 350 nM T68251 CVH2B7 53320226 IC50 = 2800 nM T68251 CO8QK2 53320227 IC50 = 180 nM T68251 CNS3F2 53321542 IC50 = 1900 nM T68251 C4UE6R 53322469 IC50 = 30000 nM T68251 C1N2BX 53322876 IC50 = 1700 nM T68251 CSYW40 53322877 IC50 = 35000 nM T68251 CGUC59 53322878 IC50 = 2400 nM T68251 C3QHA6 53322879 IC50 = 2200 nM T68251 CI3WL5 53323418 Ki = 240 nM T68251 C0H7FQ 53324260 IC50 = 26000 nM T68251 CU7YG9 53325497 IC50 = 170 nM T68251 C4G1HK 53325498 IC50 > 9100 nM T68251 CO5L1I 53325499 IC50 = 12000 nM T68251 CZA03W 53326760 IC50 = 530 nM T68251 CM53CG 53326761 IC50 = 2500 nM T68251 CWR6T4 53326860 IC50 = 500 nM T68251 CPY02U 53327890 IC50 = 2.3 nM T68251 CPGE80 53327891 IC50 = 6 nM T68251 CLJ4G2 53328858 IC50 = 1.5 nM T68251 C4G3QL 53328859 IC50 = 2.5 nM T68251 CX1TW0 53328860 IC50 = 1.3 nM T68251 C0ZX5G 53329215 IC50 = 4 nM T68251 CSU52A 53329216 IC50 = 17 nM T68251 CHF62Q 53361485 IC50 = 140 nM T68251 CJ3F4R 53361486 IC50 = 37 nM T68251 C6Y2EV 53374826 IC50 > 100000 nM T68251 CNY03Z 53378637 Ki = 440 nM T68251 CX3DU4 53378973 Ki = 390 nM T68251 CTD1H9 53378974 Ki = 240 nM T68251 CQ04KO 53389286 IC50 = 384 nM T68251 C1IFJ8 53957122 IC50 = 210000 nM T68251 CTJ48R 54185618 IC50 = 17800 nM T68251 C24SIM 54334252 IC50 = 39 nM T68251 CSUW40 54352406 IC50 = 10 nM T68251 C7RC3A 54371779 IC50 = 10 nM T68251 C3M8GZ 54580051 IC50 = 61000 nM T68251 CL0WM9 54580052 IC50 > 10000 nM T68251 CK26XF 54580053 IC50 > 10000 nM T68251 C3LF0P 54580544 Ki = 9200 nM T68251 CA8U9V 54580837 IC50 = 4000 nM T68251 CVO09J 54581546 Ki = 110 nM T68251 CWB2Q6 54581896 IC50 = 170 nM T68251 CVK72M 54582073 IC50 = 1300 nM T68251 CBK18O 54582074 IC50 > 10000 nM T68251 CP2F1B 54582075 IC50 > 10000 nM T68251 CZNU23 54582076 IC50 > 10000 nM T68251 C0U5HZ 54582077 IC50 > 10000 nM T68251 C8SG9Y 54582079 IC50 > 10000 nM T68251 CZI6S3 54582080 IC50 = 3500 nM T68251 CD09BZ 54582543 IC50 = 1300 nM T68251 CH6Q2Z 54583016 IC50 > 10000 nM T68251 C3V9LQ 54583017 IC50 = 150 nM T68251 CT80KQ 54583018 IC50 = 620 nM T68251 CPT4L5 54583019 IC50 > 10000 nM T68251 CK52YD 54583511 Ki = 530 nM T68251 CF0SK8 54583712 IC50 = 2.5 nM T68251 CBEV27 54584024 IC50 = 3300 nM T68251 CM87DP 54584025 IC50 = 1100 nM T68251 C28GKQ 54585927 IC50 > 10000 nM T68251 CAZ76E 54586892 IC50 > 10000 nM T68251 CM0OQ3 54586893 IC50 > 10000 nM T68251 CK1NS7 54586894 IC50 > 10000 nM T68251 CMC4Y1 54586895 IC50 > 10000 nM T68251 C2MKX5 54586896 IC50 = 3800 nM T68251 CU91QP 54586897 IC50 > 10000 nM T68251 CI08RQ 54586898 IC50 = 1400 nM T68251 C6PRI4 54586899 IC50 = 7600 nM T68251 CG37UX 54587429 Ki = 430 nM T68251 CL9SC3 54587769 Ki > 40000 nM T68251 C13FSJ 54669762 Ki = 24 nM T68251 CHS01Z 54669766 Ki = 520 nM T68251 C8YLA4 54669829 IC50 = 7.5 nM T68251 C1KA8X 54669830 IC50 = 2.55 nM T68251 CZA6Q9 54669831 IC50 = 24 nM T68251 CF23NJ 54669841 IC50 = 23 nM T68251 C71KLJ 54679182 IC50 = 1260 nM T68251 CC67RV 54681831 IC50 = 610 nM T68251 C83NUI 54687474 IC50 = 9300 nM T68251 CZ6V0U 54724681 IC50 > 50000 nM T68251 CJ6HT4 54726662 IC50 = 19000 nM T68251 C9P5ES 54752445 IC50 = 0.39 nM T68251 C0HKC9 54752446 IC50 = 0.57 nM T68251 C6D9IE 54753443 IC50 = 1729.19 nM T68251 CLP2C1 54753981 IC50 = 393140 nM T68251 CQD2Z6 54757100 IC50 = 63.6 nM T68251 C7E9SG 54757202 Ki = 78000 nM T68251 CMJ90D 54757404 Ki = 62 nM T68251 CD1A3F 54757406 Ki = 69 nM T68251 C4EFI5 54757409 Ki = 420 nM T68251 C5D1TI 56649332 IC50 = 1.8 nM T68251 CGTV56 56658262 IC50 = 151600 nM T68251 C9Z4TW 56658263 IC50 = 110100 nM T68251 CAV9S4 56658410 IC50 = 42200 nM T68251 CLKA98 56659256 IC50 = 73 nM T68251 CAFN81 56659257 IC50 = 269 nM T68251 C5ATG7 56659258 IC50 = 95 nM T68251 CR0HX7 56659259 IC50 = 25 nM T68251 CI8RY0 56659946 IC50 = 249240 nM T68251 C0NK1P 56659952 IC50 = 307270 nM T68251 CL6GF3 56659954 IC50 = 166110 nM T68251 CP5K7G 56661758 IC50 = 100100 nM T68251 C1EW4P 56661759 IC50 = 105600 nM T68251 C5FR4E 56661895 IC50 = 119500 nM T68251 CG7E1O 56662736 IC50 = 13 nM T68251 CZF86Q 56662737 IC50 = 264 nM T68251 CT2G8L 56662738 IC50 = 24 nM T68251 C3LQY5 56662739 IC50 = 31 nM T68251 CQY15M 56663413 IC50 = 463380 nM T68251 CWM2L3 56663417 IC50 = 836490 nM T68251 C48JHP 56663421 IC50 = 267730 nM T68251 CIG9J2 56663694 IC50 = 1021 nM T68251 C8YPU6 56665194 IC50 = 84300 nM T68251 CV46HL 56665195 IC50 = 173100 nM T68251 C3L5SO 56665196 IC50 = 108900 nM T68251 CH4M6V 56665197 IC50 = 40600 nM T68251 C20IZG 56665371 IC50 > 1000000 nM T68251 C8ZD7Q 56666204 IC50 = 45 nM T68251 CKB12J 56666205 IC50 = 54 nM T68251 CR21IL 56666206 IC50 = 100 nM T68251 CT65HD 56666207 IC50 = 311 nM T68251 C2IVE9 56666208 IC50 = 706 nM T68251 CPM8U1 56666842 IC50 = 540030 nM T68251 CC8HS0 56669604 IC50 = 9.8 nM T68251 CLO80F 56669605 IC50 = 60 nM T68251 CPS48C 56669606 IC50 = 329 nM T68251 CGMF96 56669607 IC50 = 47 nM T68251 CG0N1D 56670269 IC50 = 251910 nM T68251 CD1UX2 56670273 IC50 = 276440 nM T68251 C6O4TD 56672133 IC50 > 1000000 nM T68251 CRZF93 56672134 IC50 = 157400 nM T68251 C5C3OA 56672135 IC50 = 149200 nM T68251 CSU81T 56672275 IC50 = 133800 nM T68251 CBX8M4 56673120 IC50 = 15 nM T68251 C6Z7VA 56673121 IC50 = 86 nM T68251 C2YJZ8 56673122 IC50 = 2.9 nM T68251 C3BD9S 56673123 IC50 = 264 nM T68251 CG10FP 56673124 IC50 = 681 nM T68251 CMNQ68 56673125 IC50 = 20 nM T68251 CY80GQ 56673788 IC50 = 656770 nM T68251 C8C3QL 56675664 IC50 = 111300 nM T68251 CWI28X 56676443 IC50 = 16 nM T68251 CSPX53 56676444 IC50 = 22 nM T68251 CJU1M7 56676445 IC50 = 16 nM T68251 CGD90C 56676446 IC50 = 268 nM T68251 CCA39I 56676447 IC50 = 83 nM T68251 CL67JD 56677116 IC50 = 516830 nM T68251 CWH5R6 56677118 IC50 = 939570 nM T68251 CX80RM 56677120 IC50 = 157420 nM T68251 CKLQ67 56678865 IC50 = 67400 nM T68251 C3ZAX6 56678866 IC50 = 44100 nM T68251 C2M1TR 56678867 IC50 = 119300 nM T68251 CNE08Y 56678974 IC50 = 40400 nM T68251 C7G9AH 56678975 IC50 = 94000 nM T68251 C02GOU 56679764 IC50 = 9.4 nM T68251 CFDR70 56679765 IC50 = 13 nM T68251 CLPF34 56679766 IC50 = 29 nM T68251 C0XP1D 56679767 IC50 = 50 nM T68251 CTE68Z 56679768 IC50 = 30 nM T68251 CES0V3 56679769 IC50 = 411 nM T68251 C0L2JS 56682178 IC50 = 61300 nM T68251 C8UB9G 56682179 IC50 = 83900 nM T68251 C4XL3Y 56682293 IC50 = 86600 nM T68251 CK70XW 56682294 IC50 = 107100 nM T68251 C67VUX 56682295 IC50 = 52700 nM T68251 CIB34L 56683087 IC50 = 10 nM T68251 CM79IH 56683088 IC50 = 1.1 nM T68251 CSL1X7 56683089 IC50 = 104 nM T68251 CSR32E 56683090 IC50 = 86 nM T68251 CWJ65H 56683091 IC50 = 308 nM T68251 CEO93F 56683092 IC50 = 106 nM T68251 CO8FP7 56683093 IC50 = 80 nM T68251 C6KT1Z 56683094 IC50 = 25 nM T68251 CJCI10 56683095 IC50 = 54 nM T68251 C5F7WT 56683096 IC50 = 142 nM T68251 C62FZC 56835063 IC50 = 501 nM T68251 CKJ9S1 56835167 IC50 = 30 nM T68251 C21CLZ 56835168 IC50 = 240 nM T68251 C0L2TS 56835169 IC50 = 1200 nM T68251 CKEV19 56850269 IC50 > 500000 nM T68251 C13DBR 56850270 IC50 > 500000 nM T68251 C05CTJ 56850271 IC50 = 30000 nM T68251 CX8QD5 56850272 IC50 = 310000 nM T68251 C1I9RE 56850407 IC50 > 500000 nM T68251 CVJ90W 56850408 IC50 = 24000 nM T68251 CPI5G0 56850409 IC50 = 83000 nM T68251 C8TH2F 56945850 IC50 = 203 nM T68251 CD72TG 56945851 IC50 = 5 nM T68251 C8J4SC 56945854 IC50 = 64 nM T68251 C1AIZ6 56945963 IC50 = 29 nM T68251 CXQC91 56945964 IC50 = 58 nM T68251 CM4H9D 56945965 IC50 = 44 nM T68251 CUT4S2 56946063 IC50 = 202 nM T68251 C2CQR8 56946064 IC50 = 22 nM T68251 C2H8PG 56946065 IC50 = 13 nM T68251 CW2P6A 56946167 IC50 = 12 nM T68251 CT8S3G 56946168 IC50 = 52 nM T68251 C6LR7O 56964014 IC50 = 328 nM T68251 CE12KU 56964015 IC50 = 158 nM T68251 CL42CX 56964110 IC50 = 219 nM T68251 C0KPD8 57384084 IC50 = 9 nM T68251 CV67JB 57384091 IC50 = 53 nM T68251 C5WFN6 57391082 IC50 = 1 nM T68251 C9BN4F 57391101 IC50 = 7 nM T68251 CI0X9S 57391136 IC50 = 10 nM T68251 CD9J1C 57391201 IC50 > 10000 nM T68251 CN2H9K 57391204 IC50 = 5011.87 nM T68251 CR8MW2 57391205 IC50 = 5011.87 nM T68251 CA25DM 57391224 IC50 = 200 nM T68251 C6P9XK 57391225 IC50 = 144 nM T68251 COT76D 57391411 IC50 > 500000 nM T68251 CJZ0U8 57391412 IC50 > 500000 nM T68251 CAQB32 57391413 IC50 = 4000 nM T68251 CCB9H2 57391414 IC50 = 9 nM T68251 CC57MO 57392866 IC50 = 3.7 nM T68251 C4IWN7 57392867 IC50 = 85 nM T68251 C1ZG3T 57392880 IC50 = 2 nM T68251 CH1I4N 57392901 IC50 = 102 nM T68251 C7CV1B 57392902 IC50 = 6913 nM T68251 C25FAK 57392903 IC50 = 16 nM T68251 C4CK0Q 57392968 IC50 = 7943.28 nM T68251 CNQ9B2 57392969 IC50 = 19952.62 nM T68251 CTYP14 57392972 IC50 = 7943.28 nM T68251 C5VB0U 57392973 IC50 = 6309.57 nM T68251 CMQL31 57392974 IC50 > 10000 nM T68251 C39OHF 57392975 IC50 = 7943.28 nM T68251 CX89EL 57392993 IC50 = 607 nM T68251 C0F3ZD 57393177 IC50 > 500000 nM T68251 CUJD65 57393178 IC50 = 400000 nM T68251 CMB13S 57393179 IC50 = 9000 nM T68251 CJ30LT 57393180 IC50 = 340000 nM T68251 CT2E8Z 57393181 IC50 = 31000 nM T68251 C2O9QP 57394596 IC50 = 2 nM T68251 CN9X5F 57394606 IC50 = 2 nM T68251 CP5BX6 57394607 IC50 = 3.9 nM T68251 CA09RY 57394649 IC50 = 197 nM T68251 CDCW73 57394678 IC50 > 500000 nM T68251 CH6BA3 57394709 IC50 > 10000 nM T68251 CNOH63 57394711 IC50 = 7300 nM T68251 C1CYK9 57394729 IC50 = 25 nM T68251 C9JC3H 57394730 IC50 = 200 nM T68251 C80FML 57394731 IC50 = 111 nM T68251 CYFJ06 57394732 IC50 = 3286 nM T68251 CE5X3D 57394850 IC50 = 10 nM T68251 C82ATC 57394900 IC50 = 3000 nM T68251 C2X8UO 57394901 IC50 > 500000 nM T68251 CN8A6U 57394902 IC50 = 330000 nM T68251 CG43ME 57394903 IC50 = 13 nM T68251 C18PVK 57396348 IC50 > 1000 nM T68251 CM8K2T 57396360 IC50 > 1000 nM T68251 COXA03 57396390 IC50 = 308 nM T68251 CO17CH 57396398 IC50 = 306 nM T68251 CDES09 57396473 IC50 = 1995.26 nM T68251 CONH52 57396474 IC50 = 7943.28 nM T68251 CV51ME 57396475 IC50 = 6309.57 nM T68251 CJB27Z 57396489 IC50 = 81 nM T68251 C34RZI 57396490 IC50 = 178 nM T68251 CD5G3V 57396665 IC50 > 500000 nM T68251 CEB81P 57396666 IC50 > 500000 nM T68251 CMNU14 57396667 IC50 > 500000 nM T68251 CN0LI1 57396668 IC50 = 710 nM T68251 C2MI0H 57398136 IC50 = 1599 nM T68251 C98EXD 57398159 IC50 = 3 nM T68251 C1BIM8 57398160 IC50 = 11 nM T68251 C0KPT7 57398161 IC50 = 2.4 nM T68251 CD6Q9F 57398187 IC50 = 163 nM T68251 CSX81J 57398194 IC50 = 1610 nM T68251 CBH82N 57398195 IC50 = 45 nM T68251 C0YHM7 57398273 IC50 = 83 nM T68251 C5R1PU 57398274 IC50 = 3670 nM T68251 C0ZL1D 57399843 IC50 = 2050 nM T68251 CI6WB3 57399844 IC50 = 30083 nM T68251 C5SVE2 57399911 IC50 > 10000 nM T68251 CZ4GX2 57399912 IC50 = 7943.28 nM T68251 C4J5LE 57399913 IC50 = 7943.28 nM T68251 CH1J9Q 57399914 IC50 > 10000 nM T68251 CD50CO 57399918 IC50 = 3981.07 nM T68251 C82HGR 57399936 IC50 = 4370 nM T68251 CAX15U 57399937 IC50 = 9200 nM T68251 C1CN3U 57401566 IC50 = 2319 nM T68251 C3EKY4 57401585 IC50 = 4 nM T68251 CBZ36R 57401604 IC50 = 3 nM T68251 CM9D3A 57401688 IC50 > 10000 nM T68251 CF02UP 57401689 IC50 = 3981.07 nM T68251 CVO56U 57401690 IC50 = 7943.28 nM T68251 CN27EP 57401691 IC50 = 6309.57 nM T68251 CJLZ14 57401692 IC50 > 10000 nM T68251 C2AI8P 57401693 IC50 > 10000 nM T68251 CLNT30 57401717 IC50 = 798 nM T68251 CKL68A 57401718 IC50 = 307 nM T68251 C5IYO8 57401900 IC50 > 500000 nM T68251 CI1ML6 57401901 IC50 > 500000 nM T68251 C2IE0C 57401902 IC50 = 6800 nM T68251 C39ELP 57403329 IC50 = 15 nM T68251 CWP09F 57403330 IC50 > 1000 nM T68251 CIB91W 57403331 IC50 = 0.55 nM T68251 C63WPS 57403332 IC50 = 0.49 nM T68251 CXF62Z 57403333 IC50 = 16 nM T68251 CT26AL 57403355 IC50 = 931 nM T68251 C6OQH8 57403420 IC50 = 1258.93 nM T68251 C2Z6EC 57403421 IC50 = 5011.87 nM T68251 CA5Z2V 57403422 IC50 = 6309.57 nM T68251 CK68EY 57403424 IC50 = 7943.28 nM T68251 CQN8L6 57403445 IC50 = 232 nM T68251 C2L1SE 57403446 IC50 = 180 nM T68251 C0G2VY 57403564 IC50 = 0.8 nM T68251 CK4CJ0 57403617 IC50 = 290000 nM T68251 C5D0WE 57403618 IC50 > 500000 nM T68251 C7K2AP 57403619 IC50 > 500000 nM T68251 CE9B2P 57403620 IC50 = 1700 nM T68251 C1DRY0 57403621 IC50 = 200 nM T68251 C2MH8O 57523473 IC50 = 0.35 nM T68251 C57CEM 57523505 IC50 = 4 nM T68251 CS8W4L 57523538 IC50 = 5 nM T68251 CIT7B9 57523539 IC50 = 2 nM T68251 C56QXU 57523540 IC50 = 4 nM T68251 CX8IU3 57523541 IC50 = 30 nM T68251 CE8CL9 57523575 IC50 = 107 nM T68251 CWUP89 57523576 IC50 = 0.13 nM T68251 CT2QS3 57523577 IC50 = 0.07 nM T68251 CK6M0Y 57523578 IC50 = 0.1 nM T68251 C0HVU7 57523611 IC50 = 3 nM T68251 C5Q0ND 57523641 IC50 = 1.2 nM T68251 CWH7V8 57561293 IC50 = 533 nM T68251 C1PHI6 57708731 IC50 = 510 nM T68251 CF2Z7W 57708783 IC50 = 62 nM T68251 C9KV2W 57708792 IC50 = 660 nM T68251 CE36GP 57708799 IC50 = 670 nM T68251 C23QGY 57708843 IC50 > 1000 nM T68251 C2J5CW 57708880 IC50 = 230 nM T68251 C1K6AP 57708886 IC50 = 14 nM T68251 CY1N3J 57792153 IC50 = 1167 nM T68251 C6BKQ0 57874709 IC50 = 46000 nM T68251 CCKD80 58307579 Ki = 2.3 nM T68251 CX73PT 59033102 IC50 > 25000 nM T68251 CAT67H 59910477 IC50 = 79 nM T68251 CTZJ24 59910497 IC50 = 885 nM T68251 C1T2QI 60144811 IC50 = 545000 nM T68251 CZ18UT 67684770 IC50 = 10700 nM T68251 CLOE02 70682288 Ki = 600 nM T68251 CH2Q3V 70682301 IC50 = 53 nM T68251 C4NG7I 70682302 IC50 = 24 nM T68251 C6YOW4 70682303 IC50 = 10 nM T68251 CH76IU 70684364 Ki = 450 nM T68251 CZ63AG 70684365 Ki = 300 nM T68251 C6YH8C 70684382 IC50 = 3.8 nM T68251 CQ50YR 70684390 IC50 = 66 nM T68251 CTR64D 70686538 IC50 = 149 nM T68251 C0Q6JA 70686539 IC50 = 179 nM T68251 C8B6WD 70688393 IC50 = 11650 nM T68251 CGR3J2 70688394 IC50 = 23280 nM T68251 CTUN76 70688632 Ki = 61 nM T68251 C3LCG0 70688633 Ki = 180 nM T68251 CV9Y7S 70688643 IC50 = 7.3 nM T68251 CB4ZL3 70690154 IC50 > 500000 nM T68251 CJY19I 70690714 IC50 = 15 nM T68251 CFM0Q5 70690777 IC50 = 0.2 nM T68251 CWVI71 70691250 IC50 = 144 nM T68251 CJ3OY4 70692312 IC50 > 500000 nM T68251 C1A0VU 70692840 Ki = 110 nM T68251 CY4E9Z 70692916 IC50 > 100000 nM T68251 C0HFX4 70694371 IC50 > 500000 nM T68251 C0HE2P 70694634 IC50 = 15470 nM T68251 CLE79H 70696450 IC50 > 500000 nM T68251 CENQ98 70697478 IC50 = 450 nM T68251 C1XNI9 70941086 IC50 > 100000 nM T68251 C7BHO9 70941091 IC50 = 34700 nM T68251 C37VPQ 70941121 IC50 = 10300 nM T68251 CF7PC5 70941155 IC50 > 100000 nM T68251 CL7JF9 71304794 IC50 = 63 nM T68251 CSY30R 71304795 IC50 = 10 nM T68251 CNPG78 71304796 IC50 = 170 nM T68251 CA92XR 71449332 IC50 = 85500 nM T68251 COM1B0 71449369 IC50 = 143 nM T68251 CA6IB0 71450469 IC50 > 1000000 nM T68251 CK2AT8 71451145 IC50 = 12500 nM T68251 C5NYF7 71451146 IC50 = 1400 nM T68251 CW06TJ 71451147 IC50 = 67 nM T68251 CA7M9F 71451166 IC50 = 39000 nM T68251 CD4CP2 71451167 IC50 = 60000 nM T68251 C6M9VL 71451168 IC50 = 8100 nM T68251 C7HUF5 71451169 IC50 = 120 nM T68251 CMW3O0 71451330 Ki > 200000 nM T68251 CT5J7F 71452300 IC50 > 1000000 nM T68251 C23NVO 71452301 IC50 > 1000000 nM T68251 C7UIS9 71452970 IC50 = 67500 nM T68251 CC1B0Z 71452971 IC50 = 83700 nM T68251 CNMP23 71452972 IC50 = 27600 nM T68251 CIP9J5 71452973 IC50 = 8100 nM T68251 CUZ9S0 71452974 IC50 = 120 nM T68251 C71TWC 71452975 IC50 = 3900 nM T68251 CE98YL 71452999 IC50 = 184 nM T68251 C8VC6N 71453000 IC50 = 30 nM T68251 C4VKI1 71453001 IC50 = 87 nM T68251 C4E6PS 71453593 IC50 = 20000 nM T68251 C5K8WS 71454094 IC50 = 573000 nM T68251 CP2D3C 71454095 IC50 > 1000000 nM T68251 CGE27K 71454723 IC50 = 3000 nM T68251 C3VQW4 71455829 IC50 > 1000000 nM T68251 C4EJX2 71456472 IC50 = 37 nM T68251 C9QS6E 71456659 Ki = 20 nM T68251 C1JI6W 71458326 IC50 = 74600 nM T68251 C8ZR2I 71458327 IC50 = 1700 nM T68251 CV2J5Y 71458328 IC50 = 460 nM T68251 C29YHS 71458330 IC50 = 900 nM T68251 CXC1U7 71458350 IC50 = 121 nM T68251 C4IZ5V 71458351 IC50 = 181 nM T68251 CKR4D0 71459517 IC50 > 1000000 nM T68251 CKV4Q6 71460169 IC50 = 4500 nM T68251 CYF62U 71460170 IC50 = 750 nM T68251 C3LFX2 71460171 IC50 = 270 nM T68251 CDRO30 71460172 IC50 = 25 nM T68251 C6WN3A 71460173 IC50 = 13 nM T68251 CZO86D 71460193 IC50 = 278 nM T68251 C6UQW4 71461261 IC50 > 1000000 nM T68251 CKW27N 71461578 IC50 = 19.6 nM T68251 CX7W4A 71461879 IC50 = 2400 nM T68251 CKXO81 71461880 IC50 = 6300 nM T68251 CI4M8V 71461881 IC50 = 7600 nM T68251 CHD70Q 71461882 IC50 = 29 nM T68251 C7MLC8 71461883 IC50 = 17 nM T68251 CWL97M 71461905 IC50 = 301 nM T68251 CUT3H5 71461906 IC50 = 148 nM T68251 C06AXC 71461907 IC50 = 58 nM T68251 CSW59Y 71461908 IC50 = 1340 nM T68251 C9QE5X 71462985 IC50 > 1000000 nM T68251 CATP87 71465323 IC50 = 32.8 nM T68251 C0H3BX 71465324 IC50 = 6.4 nM T68251 CTM24Y 71465370 IC50 = 7.2 nM T68251 C6ZV0X 71465371 IC50 = 9.3 nM T68251 C7NYO8 71465420 IC50 = 6.3 nM T68251 C0E3FD 71465421 IC50 = 3.9 nM T68251 CW1K8M 71465466 IC50 > 100000 nM T68251 C28OYX 71465467 IC50 = 35700 nM T68251 C12BUO 71465468 IC50 > 100000 nM T68251 CP37ZB 71465510 IC50 = 2100 nM T68251 CR2T8F 71503450 IC50 = 2.8 nM T68251 C56YRV 71516803 IC50 < 1 nM T68251 C52QIK 71516804 IC50 = 5.1 nM T68251 C79ZRK 71516805 IC50 = 1.6 nM T68251 C3L7SD 71533484 IC50 = 227 nM T68251 CZH5S9 71533485 IC50 = 52 nM T68251 C4YRC7 71533486 IC50 = 21 nM T68251 CGM72Q 71540498 IC50 = 57 nM T68251 CXA1I5 71540599 IC50 = 54 nM T68251 C7CV9E 71540600 IC50 = 149 nM T68251 CA4BP6 71540601 IC50 = 82 nM T68251 CMZ3T2 71540715 IC50 = 67 nM T68251 CXY83G 71540716 IC50 = 56 nM T68251 C1ZH2G 71540717 IC50 = 69 nM T68251 CT4UD5 71540831 IC50 = 145 nM T68251 CP7SX8 71540832 IC50 = 71 nM T68251 C9IW7R 71540833 IC50 = 54 nM T68251 C6MA8T 71540949 IC50 = 598 nM T68251 C52FXB 71547352 IC50 = 1.7 nM T68251 C9RE0A 71559535 IC50 = 8.44 nM T68251 C47TMN 71559652 IC50 = 8.46 nM T68251 CN2XB4 71559653 IC50 = 5.57 nM T68251 CZHQ79 71559654 IC50 = 1524.69 nM T68251 CO59LK 71559762 IC50 = 4.18 nM T68251 CGL35Z 71559763 IC50 = 5.62 nM T68251 C7U5LE 71559764 IC50 = 1674.81 nM T68251 CD6L1J 71559765 IC50 = 4.32 nM T68251 CXKO04 71559766 IC50 = 5.73 nM T68251 CA14SK 71559767 IC50 = 1724.94 nM T68251 COZ56A 71559768 IC50 = 9.09 nM T68251 CZ9X1J 71559769 IC50 = 1867.71 nM T68251 C5NHI1 71559770 IC50 = 8.59 nM T68251 CF9JE8 71559897 IC50 = 9.11 nM T68251 CGT96R 71559898 IC50 = 5.47 nM T68251 C01PTX 71559899 IC50 = 1674.23 nM T68251 C96OCB 71559900 IC50 = 5.53 nM T68251 CJB0D9 71559901 IC50 = 1764.37 nM T68251 C6Y1IE 71559902 IC50 = 4.09 nM T68251 C24ZYC 71559903 IC50 = 5.62 nM T68251 CC3MY7 71559904 IC50 = 1754.54 nM T68251 C7WMU5 71560026 IC50 = 9.01 nM T68251 C60VEX 71560027 IC50 = 1578.64 nM T68251 CN1VF7 71560028 IC50 = 8.39 nM T68251 CSY3D5 71560029 IC50 = 9.04 nM T68251 CH5J4A 71602247 IC50 = 16 nM T68251 CH53IU 71602248 IC50 = 230 nM T68251 C97EWQ 71602249 IC50 = 61 nM T68251 CNX9B1 71652215 IC50 = 1.4 nM T68251 C7RZN9 71652216 IC50 = 3.8 nM T68251 C0NTU7 71652382 IC50 = 0.43 nM T68251 CA5XS1 71652383 IC50 = 46 nM T68251 CYS46I 71652677 IC50 = 3200 nM T68251 CX67VE 71654516 IC50 = 3000 nM T68251 C6KEH0 71680708 Ki = 27 nM T68251 C7DMX5 71680709 Ki = 3.9 nM T68251 CFPM82 71680710 Ki = 35 nM T68251 C9ZOM7 71680866 Ki = 3.1 nM T68251 CQ68LT 71680868 Ki = 7000 nM T68251 CFH2V0 71681183 Ki = 49 nM T68251 CV3X1T 71682766 Ki = 810 nM T68251 C5EAO8 71682767 Ki = 430 nM T68251 C80EYX 71682913 Ki = 7200 nM T68251 CIBD03 71682914 Ki = 240 nM T68251 C41BYG 71682915 Ki = 4.6 nM T68251 C93XEI 71682916 Ki = 67 nM T68251 CQ29PJ 71682917 Ki = 50000 nM T68251 CFWN65 71683062 Ki = 5700 nM T68251 CM4E5A 71716445 IC50 = 4.19 nM T68251 C45PSZ 71717046 IC50 = 9.26 nM T68251 C9Z4PI 71718276 IC50 = 8.41 nM T68251 C2XW5I 71718291 IC50 = 9.41 nM T68251 C3L4XU 71718301 IC50 = 3.3 nM T68251 C18RDB 71719502 IC50 = 4.43 nM T68251 C6FVE5 71734008 IC50 < 1 nM T68251 CN95PL 71734104 IC50 < 1 nM T68251 CV37BJ 71734105 IC50 = 4.8 nM T68251 C7H8VM 71734106 IC50 < 1 nM T68251 CHBV73 71734107 IC50 < 1 nM T68251 C6C1JF 71734108 IC50 = 14 nM T68251 CR28AW 71734195 IC50 = 7 nM T68251 C2YJR3 71734196 IC50 = 141 nM T68251 CJC6N5 71734197 IC50 = 5.2 nM T68251 CEF50T 71734198 IC50 = 3.6 nM T68251 CLWC38 72193198 IC50 < 1 nM T68251 CX4G0R 72204928 IC50 = 28200 nM T68251 CG9C6U 72204929 IC50 = 6000 nM T68251 C5A6XZ 72204930 IC50 = 20000 nM T68251 C0XZK4 72204931 IC50 = 15000 nM T68251 CM8Y7X 72204932 IC50 = 36000 nM T68251 C6RY4X 72204933 IC50 = 6600 nM T68251 C4N5AB 72204934 IC50 = 20800 nM T68251 C3H2FZ 72205111 IC50 = 42000 nM T68251 CQ0VX7 72205112 IC50 = 25000 nM T68251 CQ7TI1 72205113 IC50 = 2800 nM T68251 CPAW52 72205114 IC50 = 2100 nM T68251 C2LD3J 72205115 IC50 = 2800 nM T68251 CE4J8F 72711063 Ki = 290 nM T68251 CW2RF1 72711064 Ki = 490 nM T68251 CC5T1Q 72711065 Ki = 680 nM T68251 C7YFC8 72711513 IC50 = 1045 nM T68251 CTM4P2 72713638 IC50 = 1.2 nM T68251 C0N2JX 72713639 IC50 = 3 nM T68251 CF4K8Y 72713862 IC50 = 7.5 nM T68251 C3R6JO 72713863 IC50 = 48 nM T68251 CW9D3V 72713864 IC50 = 15 nM T68251 CQ6FH3 72713865 IC50 = 7.8 nM T68251 C4FYB0 72713866 IC50 = 20 nM T68251 CH6SI1 72713867 IC50 = 41 nM T68251 CS21QM 72713868 IC50 = 670 nM T68251 CB56AP 72714081 IC50 = 18 nM T68251 C1CK0E 72714082 IC50 = 1750 nM T68251 CP5Q8W 72714083 IC50 = 1870 nM T68251 CA03NU 72714084 IC50 = 125000 nM T68251 CRUH64 72714085 IC50 = 3800 nM T68251 COQZ24 72714091 Ki = 160 nM T68251 CC0ZX4 72714092 Ki = 230 nM T68251 CW8I1S 72714093 Ki = 310 nM T68251 C3Q9LV 72714094 Ki = 480 nM T68251 CZFY06 72714322 IC50 = 4100 nM T68251 CDY70J 72714323 IC50 = 1440 nM T68251 CD56BA 72714324 IC50 = 240 nM T68251 CE51LQ 72714333 Ki = 550 nM T68251 CK6D5F 72714334 Ki = 760 nM T68251 C1R2UZ 72714335 Ki = 690 nM T68251 CH4VF7 72714336 Ki = 440 nM T68251 C4VSK6 72714337 Ki = 560 nM T68251 CG4KW2 72714338 Ki = 420 nM T68251 C9FL7V 72714339 Ki = 50 nM T68251 CT5U1W 72734852 IC50 = 428990 nM T68251 C4OEI9 72734853 IC50 = 20620 nM T68251 C4AT5M 72734854 IC50 = 6559 nM T68251 CA7I9Q 72734855 IC50 = 10800 nM T68251 CJ5N2K 72734856 IC50 = 679 nM T68251 CCQ27I 72734857 IC50 = 1802 nM T68251 CCP65R 72735032 IC50 = 5438 nM T68251 C5XL1A 72735033 IC50 = 386 nM T68251 CYT1H0 72735034 IC50 = 530 nM T68251 CW6IE4 72735035 IC50 = 325 nM T68251 C58RHN 72735036 IC50 = 678.1 nM T68251 CFB5U1 72735037 IC50 = 325 nM T68251 CXY79G 72737387 IC50 = 2776 nM T68251 C6M1OD 72737388 IC50 = 834.9 nM T68251 CY4M3X 72737389 IC50 = 28190 nM T68251 CQM2E0 72737390 IC50 = 9480 nM T68251 CFQX60 72737391 IC50 = 878 nM T68251 C4BAJ5 72737560 IC50 = 77930 nM T68251 CRP56E 72737561 IC50 = 3093 nM T68251 C3J8GN 72737562 IC50 = 7480 nM T68251 CS2JM8 72737563 IC50 = 678 nM T68251 CZ0G7Y 72737564 IC50 = 786 nM T68251 COHR84 72737565 IC50 = 877 nM T68251 CLV1F5 72737566 IC50 = 516 nM T68251 CDX2F9 72984326 IC50 = 9.25 nM T68251 C6SR0A 73106454 IC50 = 61.94 nM T68251 CUKG79 73292708 IC50 = 0.9 nM T68251 C5D3CJ 73292709 IC50 = 4 nM T68251 CL69NM 73292710 IC50 = 4 nM T68251 CQ4RO1 73292711 IC50 = 0.7 nM T68251 C7CT2E 73292869 IC50 = 4 nM T68251 CA0LS6 73292870 IC50 = 0.9 nM T68251 CJU3V6 73292871 IC50 = 5 nM T68251 C3PGF2 73292872 IC50 = 3 nM T68251 C0O8VM 73292873 IC50 = 2 nM T68251 CBR9I5 73293034 IC50 = 3 nM T68251 C9FD2C 73293035 IC50 = 3 nM T68251 C7LP5J 73293036 IC50 = 2 nM T68251 C9PQG1 73293037 IC50 = 5 nM T68251 C4PF1H 73293038 IC50 = 0.4 nM T68251 CE39WF 73293196 IC50 = 4 nM T68251 CU96XE 73293197 IC50 = 9 nM T68251 CGC51Z 73293198 IC50 = 2 nM T68251 CC83FW 73293199 IC50 = 2 nM T68251 CS6T8M 73293200 IC50 = 0.5 nM T68251 C38IDL 73345835 Ki = 1.7 nM T68251 CR1LT3 73346934 IC50 = 200630 nM T68251 C25SOB 73349251 IC50 = 0.8 nM T68251 CW01EA 73349535 IC50 > 10000 nM T68251 C8ROG3 73350414 Ki = 14 nM T68251 CF7AB2 73350415 Ki = 17 nM T68251 C2PFM4 73351930 Ki = 200 nM T68251 COC60V 73352986 IC50 = 671560 nM T68251 CI09CY 73354906 Ki = 8.5 nM T68251 CA5T7P 73603957 IC50 = 3000 nM T68251 C8VN1R 74221194 IC50 = 1800 nM T68251 C7M4FT 74430862 IC50 = 35670 nM T68251 CD28XO 74966628 IC50 = 109.9 nM T68251 CG1AU5 74991907 IC50 = 2.6 nM T68251 C65RFS 74991938 IC50 = 6.6 nM T68251 CX89MG 75002237 IC50 = 34197.94 nM T68251 CD7P3T 75002250 IC50 = 750 nM T68251 CU73SM 75018048 IC50 = 26 nM T68251 C1BTU7 75018058 IC50 = 29.99 nM T68251 CX9VB7 75018063 IC50 = 15 nM T68251 CLHO50 75018065 IC50 = 3.396 nM T68251 CQL0E1 75018100 IC50 = 1 nM T68251 CC9UA2 75018101 IC50 = 1.3 nM T68251 CYB42V 75018103 IC50 = 269.77 nM T68251 C1FTQ8 75018104 IC50 = 5.8 nM T68251 C5M2FT 75018105 IC50 = 1.6 nM T68251 CF5ZC7 75018120 IC50 = 50 nM T68251 CFW35X 75018121 IC50 = 280 nM T68251 C4GK3X 75018123 IC50 = 5105.05 nM T68251 C6FPO0 75018124 IC50 = 84 nM T68251 CMS1L6 75018126 IC50 = 3500 nM T68251 CW78YB 75018133 IC50 = 38.02 nM T68251 CZP6X1 75018134 IC50 = 414 nM T68251 CS1D6P 75018135 IC50 = 0.4 nM T68251 CHAP32 75018146 IC50 = 2430 nM T68251 CEF3L5 75018147 IC50 = 6.397 nM T68251 CPMC39 75018148 IC50 = 779.83 nM T68251 CBNW85 75018149 IC50 = 53.95 nM T68251 C57SNU 75018158 IC50 = 309.74 nM T68251 CCL95X 75018159 IC50 = 33.96 nM T68251 CXC24A 75018160 IC50 = 210 nM T68251 C9F8BU 75018162 IC50 = 920 nM T68251 C4OP3D 75018163 IC50 = 100 nM T68251 C7YPR3 75018171 IC50 = 51999.6 nM T68251 CT8Y6H 75018172 IC50 = 1698.24 nM T68251 C5Z1CN 75018180 IC50 = 1 nM T68251 CW7OX3 75018184 IC50 = 6800 nM T68251 C68QBF 75018185 IC50 = 10.99 nM T68251 CSBO46 75018194 IC50 = 41 nM T68251 CUB7V9 76329513 IC50 = 0.26 nM T68251 C5LB0U 78426619 IC50 > 100000 nM T68251 CET6N8 78426757 IC50 > 100000 nM T68251 CKD41G 81689861 IC50 = 1000 nM T68251 CBL02O 85040463 IC50 = 27.99 nM T68251 CHAG58 85052312 IC50 = 6.6 nM T68251 CJ67RP 85055259 IC50 = 59 nM T68251 CVHM18 85082338 IC50 = 11.99 nM T68251 CRC43U 85102289 IC50 = 0.4 nM T68251 C3Z0PJ 85141621 IC50 = 0.2 nM T68251 C28SQI 85198610 IC50 = 11 nM T68251 CUE7G4 86287514 IC50 = 24000 nM T68251 CGQ8F3 86287515 IC50 = 1800 nM T68251 CJ37XE 86287516 IC50 = 3200 nM T68251 COV8I9 86291010 IC50 = 1088 nM T68251 C76RBA 86298624 IC50 = 230 nM T68251 C93FKI 86298625 IC50 = 110 nM T68251 CVLU48 86298626 IC50 = 192 nM T68251 CAB2F5 87349434 Ki = 13000 nM T68251 CY74HT 89136066 IC50 = 2 nM T68251 C1MDQ8 89136114 IC50 = 1400 nM T68251 CO2FL5 90137145 IC50 = 310 nM T68251 CIJ96H 90644155 IC50 = 4800 nM T68251 CX7EW1 90644156 IC50 = 30000 nM T68251 CK5GZ4 90644157 IC50 = 52000 nM T68251 C7O1YN 90644158 IC50 = 19000 nM T68251 CEN6C1 90644159 IC50 = 4900 nM T68251 C8X9UZ 90644160 IC50 = 16000 nM T68251 C3H6SG 90656558 IC50 = 980 nM T68251 CFE10C 90656560 IC50 = 1030 nM T68251 CD4L8R 90656562 IC50 = 4190 nM T68251 CEST81 90656564 IC50 = 2710 nM T68251 C7J0CO 90656566 IC50 = 520 nM T68251 CE9Y4D 90656568 IC50 = 1940 nM T68251 CZVG63 90656570 IC50 = 720 nM T68251 CT0QG6 90656572 IC50 = 760 nM T68251 CFPR48 90656574 IC50 = 3360 nM T68251 CDF06N 90656576 IC50 = 1810 nM T68251 CQ3R1A 90656578 IC50 = 270 nM T68251 CWV0Z9 90656580 IC50 = 1280 nM T68251 CGX01J 90656582 IC50 = 430 nM T68251 C6M1VH 90656584 IC50 = 26180 nM T68251 C1GUD2 90656586 IC50 = 38320 nM T68251 C5KWT1 90656588 IC50 = 7430 nM T68251 CS7PZ6 90656590 IC50 = 5760 nM T68251 CGF9P3 90656592 IC50 = 1520 nM T68251 CM46JO 90656594 IC50 = 5210 nM T68251 CXL84V 90656596 IC50 = 2070 nM T68251 C7EIO6 90656598 IC50 = 2320 nM T68251 CRH7F2 90656600 IC50 = 4360 nM T68251 CKW64G 90656602 IC50 = 2950 nM T68251 C4CU3D 90656604 IC50 = 2050 nM T68251 CVPH63 90663059 Ki = 18000 nM T68251 C6AK3O 90663060 Ki = 15000 nM T68251 CUZD67 90663061 Ki = 8000 nM T68251 CTQ17J 90663062 Ki = 33000 nM T68251 CQGJ90 90663063 Ki = 6000 nM T68251 C0ZH1K 90663064 Ki = 17000 nM T68251 CD53CF 90663065 Ki = 5000 nM T68251 C1A4QT 90663067 Ki = 8000 nM T68251 CLW7Q8 90663069 Ki = 24000 nM T68251 C6JY4Q 90663070 Ki = 36000 nM T68251 C7YU1I 90663071 Ki = 10000 nM T68251 C07RTW 90663072 Ki = 11000 nM T68251 CZ68QM 90663073 Ki = 18000 nM T68251 CVTJ63 90663074 Ki = 7000 nM T68251 C9J8HB 90663075 Ki = 4000 nM T68251 C06GRV 90663076 Ki = 2000 nM T68251 CF2L9A 90663077 Ki = 40000 nM T68251 CGL0N7 90663078 Ki = 12000 nM T68251 COP05M 90663079 Ki = 13000 nM T68251 C1E5CB 90663080 Ki = 35000 nM T68251 C6IXP4 90663081 Ki = 41000 nM T68251 C0S7NT 90663082 Ki = 12000 nM T68251 C8MOY6 90663083 Ki = 20000 nM T68251 C4NP9W 90663084 Ki = 16000 nM T68251 CD3C8E 90663085 Ki = 16000 nM T68251 C63NOF 90663086 Ki = 15000 nM T68251 CU3LC2 90663087 Ki = 17000 nM T68251 CQ9C5I 90667651 IC50 = 0.53 nM T68251 CGXO89 90667652 IC50 = 0.61 nM T68251 CRT54C 101910871 IC50 = 11000 nM T68251 C1J3CK 117094707 IC50 = 5400 nM T68251 CDO15M 118721026 IC50 = 12.5 nM T68251 CHO72Q 118721027 IC50 = 1449 nM T68251 C5ZS4E 118722686 IC50 = 2100 nM T68251 CIZB24 118722687 IC50 = 6100 nM T68251 C5C0ZX 118722688 IC50 = 7100 nM T68251 C4V3FD 118723755 IC50 = 3 nM T68251 CH6OW5 122179777 IC50 = 85350 nM T68251 CLCW15 122181996 IC50 > 100000 nM T68251 CZO32N 122181998 IC50 > 100000 nM T68251 C40DWG 122181999 IC50 > 100000 nM T68251 CJFS09 122190237 IC50 = 590 nM T68251 CRN56G 122191012 IC50 = 235.2 nM T68251 CGC3E2 122191014 IC50 = 144.6 nM T68251 CS61WU 122191016 IC50 = 256.2 nM T68251 CV3SP6 122191017 IC50 = 299.2 nM T68251 C8ZOT4 122191645 IC50 = 7920 nM T68251 CU6LT0 122191646 IC50 = 2884.03 nM T68251 CER90U 122191647 IC50 = 8511.38 nM T68251 C8X2BN 122191648 IC50 = 3235.94 nM T68251 CQ3US9 122191649 IC50 = 4830 nM T68251 C86DWE 122191650 IC50 = 11220.18 nM T68251 CQ14HT 122191651 IC50 = 9430 nM T68251 C8B1HC 122191652 IC50 = 6760.83 nM T68251 CN6WP3 122191653 IC50 = 208.93 nM T68251 CJ5R2S 122192039 IC50 = 4168.69 nM T68251 CK45AP 122192040 IC50 = 794.33 nM T68251 C2W4VX 122192041 IC50 = 2700 nM T68251 C3R5YP 122192042 IC50 = 12589.25 nM T68251 C8EB9C 122192043 IC50 = 11440 nM T68251 CF2K9Z 122192044 IC50 = 14791.08 nM T68251 C68DRB 122192045 IC50 = 2089.3 nM T68251 C2L7ZO 122192046 IC50 = 2150 nM T68251 C1BH0V 122192047 IC50 = 23820 nM T68251 C9MX4H 122192048 IC50 = 17782.79 nM T68251 CE4MD1 122192049 IC50 = 15488.17 nM T68251 CU13GZ 122192050 IC50 = 2818.38 nM T68251 CN1OP2 122192051 IC50 = 9900 nM T68251 C2WV6G 122192052 IC50 = 14791.08 nM T68251 CD2I6H 122192053 IC50 = 16840 nM T68251 CQ7RZ6 122192054 IC50 = 3630.78 nM T68251 COIP89 122195564 IC50 = 360 nM T68251 C8Z1BF 124196387 IC50 = 17000 nM T68251 CF9C4N 127025165 IC50 = 6.5 nM T68251 CH59PY 127025166 IC50 = 791 nM T68251 CT03QA 127026888 IC50 = 370 nM T68251 CO1DJ9 127027301 IC50 = 11.66 nM T68251 CM7B5S 127029507 IC50 = 628 nM T68251 C6HA8I 127029508 IC50 > 100000 nM T68251 CPM3N2 127029509 IC50 = 56.3 nM T68251 C3B9EY 127029510 IC50 > 100000 nM T68251 C9NLI6 127030239 IC50 = 112260 nM T68251 CW3C0H 127030240 IC50 = 38650 nM T68251 CHC1V8 127031459 IC50 = 34790 nM T68251 C5GJB1 127031460 IC50 = 9390 nM T68251 C3R8PS 127031461 IC50 = 13220 nM T68251 C07FRX 127031462 IC50 = 90810 nM T68251 C9QC5M 127031784 IC50 = 1050 nM T68251 CX25ZP 127031785 IC50 = 210410 nM T68251 CIP36Q 127032630 IC50 = 1890 nM T68251 CA5I7G 127032946 IC50 = 410 nM T68251 CEO26U 127032998 IC50 = 28520 nM T68251 CL16WE 127033305 IC50 = 5520 nM T68251 C9RZO5 127033306 IC50 = 640 nM T68251 C20GLU 127033307 IC50 = 240 nM T68251 C2XUV8 127033875 IC50 = 74910 nM T68251 COM48Q 127033876 IC50 = 28760 nM T68251 C30DFR 127033877 IC50 = 223370 nM T68251 CA8HJ9 127033878 IC50 = 36790 nM T68251 CQ3HV1 127034380 IC50 = 566890 nM T68251 CV1YR6 127036461 IC50 = 2000 nM T68251 CDIC57 127037442 IC50 = 3 nM T68251 CV3NQ6 127037443 IC50 = 2400 nM T68251 CWI7K3 127037444 IC50 > 10000 nM T68251 C9QLI2 127037445 IC50 = 9000 nM T68251 CCA0R8 127037446 IC50 = 1100 nM T68251 C89QOM 127043503 IC50 = 51 nM T68251 CK3I0F 127043504 IC50 = 263 nM T68251 C9E5YJ 127043505 IC50 = 31 nM T68251 CW1Q3D 127043506 IC50 = 76 nM T68251 CFDC75 127043682 IC50 = 193 nM T68251 C1C7WB 127044036 IC50 = 123 nM T68251 C16UNQ 127044037 IC50 = 472 nM T68251 CN58BX 127044038 IC50 = 672 nM T68251 C5DMP0 127044039 IC50 = 419 nM T68251 CPF6U7 127044139 IC50 = 177 nM T68251 C5FPE1 127044169 IC50 > 500 nM T68251 C7YE9B 127044170 IC50 > 500 nM T68251 CT9B0Q 127044462 IC50 = 44.65 nM T68251 CL3X1A 127044649 IC50 = 98 nM T68251 C7X1YO 127044650 IC50 = 186 nM T68251 C8RZ7T 127044651 IC50 = 41 nM T68251 C3I4PT 127044652 IC50 = 103 nM T68251 CBR1V9 127044680 IC50 = 85.9 nM T68251 CDX86T 127044818 IC50 = 30 nM T68251 C56OJV 127044819 IC50 = 24 nM T68251 CF7A5N 127044986 IC50 = 843 nM T68251 CGLJ92 127045131 IC50 = 203 nM T68251 C4HY6K 127045132 IC50 = 208 nM T68251 CWO1X0 127045258 IC50 = 806 nM T68251 C43ORS 127045609 IC50 = 291 nM T68251 C21LIW 127053364 IC50 = 0.19 nM T68251 CR5VQ8 127053365 IC50 = 2.2 nM T68251 C19QXS 127053368 IC50 > 10000 nM T68251 CJ0G9N 127053369 IC50 > 10000 nM T68251 C2Q6UH 127053370 IC50 > 10000 nM T68251 CWM7U2 127053371 IC50 = 21.8 nM T68251 C1VRM8 127053372 IC50 > 10000 nM T68251 CT76DR 127053375 IC50 = 2.05 nM T68251 CYA92R 130282633 IC50 = 890 nM T68251 CO3QE2 130282636 IC50 = 1000 nM T68251 C4MB7N 132285189 Ki = 85 nM T68251 CTN42D 132941363 IC50 = 11000 nM T68251 C83FAY 134130294 Ki = 15.9 nM T68251 CT3G2U 134133460 IC50 = 0.16 nM T68251 C8VLY0 134144890 IC50 = 110 nM T68251 C93ZLI 134145328 IC50 = 107 nM T68251 CN9D7G 134155756 IC50 = 2600 nM T68251 CU24IK 134694685 IC50 = 190 nM T68251 CHV2U1 135438561 IC50 = 5300 nM T68251 C4FVJ1 135487604 IC50 = 79600 nM T68251 C6GR3K 135567051 IC50 = 83 nM T68251 C1MOD4 135567320 IC50 = 730 nM T68251 CYH23I 136054468 IC50 = 32 nM T68251 CZ8DW1 136054472 IC50 = 86 nM T68251 C9H0DL 136054473 IC50 = 120 nM T68251 CX7MI0 136054475 IC50 = 65 nM T68251 CA5JR6 136054481 IC50 = 14 nM T68251 CO2VU9 136054484 IC50 < 10 nM T68251 CV47JN 136054485 IC50 = 10 nM T68251 CZ48WO 136054487 IC50 = 23 nM T68251 CR9CY5 136054490 IC50 < 10 nM T68251 C8FGT0 136054495 IC50 = 110 nM T68251 CGH39U 136054498 IC50 < 10 nM T68251 C2TO7Y 136054508 IC50 = 160 nM T68251 CG70BZ 136054516 IC50 = 3 nM T68251 CSM57W 136054520 IC50 = 0.57 nM T68251 CXNG40 136118011 Ki = 2472 nM T68251 C1IOH9 136118012 Ki > 3333 nM T68251 CTY79S 136118013 Ki > 3333 nM T68251 CTE87J 136118014 Ki > 3333 nM T68251 CJG54U 136219136 IC50 > 30000 nM T68251 C3CAV5 136219141 IC50 > 30000 nM T68251 CPB07Z 136241630 IC50 = 800 nM T68251 CIEW62 136380958 IC50 = 8.3 nM T68251 CSEY19 137175240 IC50 = 7170 nM T68251 C9HS7J 137287436 IC50 = 1.9 nM T68251 C4UMY5 137636781 IC50 > 5000 nM T68251 CR8H9Z 137644167 IC50 > 5000 nM T68251 CB8M6U 137646865 IC50 > 5000 nM T68251 CK4LE6 137647628 IC50 = 2700 nM T68251 C9CIY6 137651719 IC50 = 2 nM T68251 CS80YI 137652598 IC50 = 280 nM T68251 CZB75K 137657128 IC50 > 10000 nM T68251 CC3I9B 137660260 IC50 > 5000 nM T68251 C4H0EM 137661370 IC50 = 3100 nM T68251 CZ8H6N 137661550 IC50 = 5800 nM T68251 C37HMX 137701229 Ki = 37 nM T68251 C5FWA2 145949488 IC50 = 584 nM T68251 CZS1N7 145949693 IC50 = 936 nM T68251 C6IPV3 145949783 IC50 = 4800 nM T68251 C72LGN 145950074 IC50 = 2850 nM T68251 CU53BP 145950331 IC50 > 5000 nM T68251 CY8C4A 145950332 IC50 = 189 nM T68251 CAJ25P 145951291 IC50 > 5000 nM T68251 C3EF7N 145952515 IC50 = 114 nM T68251 CW1GS2 145952760 IC50 > 5000 nM T68251 CFN1R7 145952843 IC50 = 187 nM T68251 CV80WQ 145954107 IC50 > 5000 nM T68251 C16VNH 145954604 IC50 = 500 nM T68251 CQF50V 145954863 IC50 = 128 nM T68251 C2HAG8 145955226 IC50 = 8520 nM T68251 CH0ZO5 145955778 IC50 = 362 nM T68251 CVZ5U7 145955868 IC50 = 232 nM T68251 C8TPR1 145956198 IC50 > 5000 nM T68251 COR96H 145956298 IC50 = 2120 nM T68251 CR8U7Y 145956318 IC50 > 5000 nM T68251 C7R3FE 145956426 IC50 = 1650 nM T68251 CUS0Y9 145957234 IC50 > 5000 nM T68251 C6MHN7 145957508 IC50 > 5000 nM T68251 CQ15DP 145957734 IC50 = 4070 nM T68251 C5K7PV 145958060 IC50 > 5000 nM T68251 CBE02W 145958354 IC50 > 5000 nM T68251 CQL4O0 145959327 IC50 > 5000 nM T68251 CG03OE 145959777 IC50 = 210 nM T68251 CIQ9J2 145960035 IC50 = 5340 nM T68251 CRY63E 145963538 IC50 > 5000 nM T68251 CX7PL8 145963779 IC50 = 75.25 nM T68251 CPRZ56 145963828 IC50 = 72.02 nM T68251 C5JTM2 145963892 IC50 = 38.68 nM T68251 CFLU54 145964255 IC50 = 57.24 nM T68251 C3MDU9 145965508 IC50 = 81210 nM T68251 C8ZI7P 145965593 IC50 = 53.14 nM T68251 C6ASH4 145965758 IC50 = 58.02 nM T68251 CABQ48 145965824 IC50 = 54.74 nM T68251 C8M7FR 145966330 IC50 = 660 nM T68251 CCO03H 145966492 IC50 = 32.71 nM T68251 CZG2P7 145966498 IC50 = 33.47 nM T68251 C4P0GM 145966951 IC50 = 53.82 nM T68251 C5ICD0 145967022 IC50 = 1350 nM T68251 CI80WY 145967366 IC50 = 19.57 nM T68251 CFE1A5 145971595 Ki = 127 nM T68251 CWY5X0 145971805 IC50 = 414 nM T68251 C1FPG2 145972660 IC50 = 219 nM T68251 CYFI60 145973042 IC50 = 2500 nM T68251 CZHR42 145973116 IC50 = 203400 nM T68251 CQF05Z 145973471 IC50 = 50.55 nM T68251 CJF73O 145973630 IC50 = 172 nM T68251 CC1BF5 145973750 IC50 = 58.08 nM T68251 COA47B 145973991 IC50 = 54.68 nM T68251 C1VO8L 145974965 IC50 = 73.82 nM T68251 CQ0DP4 145975098 IC50 = 55.13 nM T68251 CV9D1F 145975682 IC50 > 100000 nM T68251 CI9VB4 145975902 IC50 > 10000 nM T68251 CX7M9L 145976456 IC50 > 5000 nM T68251 C5C6VJ 145976464 IC50 = 54180 nM T68251 C1KPL5 145976497 IC50 = 670 nM T68251 C7RG1J 145976981 IC50 = 62.87 nM T68251 C18OCA 145976989 IC50 = 230000 nM T68251 C5HW7O 145977208 IC50 = 36.83 nM T68251 CPD1B0 145977213 IC50 > 5000 nM T68251 C79VAX 145977588 IC50 = 49.69 nM T68251 CG9KD3 145977825 IC50 > 1000 nM T68251 C60INE 145977843 IC50 = 83.04 nM T68251 CN6JB8 145978296 IC50 > 1000 nM T68251 C5Z7XW 145983264 IC50 = 182 nM T68251 C0EMZ9 145984335 IC50 = 345 nM T68251 CBNO84 145985441 IC50 = 414 nM T68251 CDW7K5 145986213 IC50 = 102 nM T68251 CM7YB8 145998092 IC50 = 1300 nM T68251 C2C8QR 153033791 IC50 = 58430 nM T68251 C2CZ9B 155511425 IC50 = 5700 nM T68251 CZ25LW 155512044 IC50 = 11000 nM T68251 CV10AF 155512426 IC50 = 151 nM T68251 C1V4CS 155512637 IC50 > 10000 nM T68251 CMQ8W6 155512861 IC50 = 7500 nM T68251 CFHU79 155514943 IC50 = 55 nM T68251 C13OQY 155515143 IC50 = 8800 nM T68251 CND4L8 155515645 IC50 = 9549.93 nM T68251 CC15YH 155515706 IC50 > 10000 nM T68251 C98HMU 155515777 IC50 = 1.2 nM T68251 C0OSL9 155516668 IC50 = 21379.62 nM T68251 C6N3DB 155517141 IC50 = 0.28 nM T68251 C3I5AL 155519394 IC50 = 6500 nM T68251 CS6ZT7 155519964 IC50 = 21 nM T68251 CG2RF3 155520398 IC50 = 2100 nM T68251 CL16UE 155520835 IC50 > 10000 nM T68251 C5C1SL 155521791 IC50 > 10000 nM T68251 C59YHT 155522902 IC50 = 503 nM T68251 C4AH9W 155525335 IC50 > 10000 nM T68251 CM9AP3 155526116 IC50 > 10000 nM T68251 C6RBG9 155527660 IC50 = 2800 nM T68251 C83IXL 155528558 IC50 = 0.16 nM T68251 CT4PA7 155528661 IC50 > 10000 nM T68251 CWB4X1 155529076 IC50 > 10000 nM T68251 CSG54J 155529234 IC50 > 10000 nM T68251 C2G0BE 155529579 IC50 > 10000 nM T68251 CC5FA9 155529859 IC50 > 10000 nM T68251 CQUA53 155531128 IC50 = 3000 nM T68251 C7TP3R 155531151 IC50 > 10000 nM T68251 CZSY48 155533962 IC50 = 3600 nM T68251 C5WTE3 155534754 IC50 = 6700 nM T68251 CG47PB 155534833 IC50 = 3000 nM T68251 C4VCN3 155535749 IC50 = 12860 nM T68251 C2WCU5 155536887 IC50 = 10715.19 nM T68251 C4DSL8 155536899 IC50 > 10000 nM T68251 C12LFZ 155540134 IC50 = 620 nM T68251 CNH2K4 155540729 IC50 = 3300 nM T68251 CO90SD 155541304 IC50 = 11748.98 nM T68251 CRY3D4 155541376 IC50 = 13 nM T68251 CV0ZI3 155542003 IC50 = 12302.69 nM T68251 CJN8X5 155542058 Ki = 0.5 nM T68251 CO8ZY9 155542845 IC50 = 0.048 nM T68251 CH9E0W 155543836 IC50 = 34673.69 nM T68251 C1VL8X 155544079 IC50 > 10000 nM T68251 CYK18P 155544623 IC50 > 10000 nM T68251 CBSJ86 155544856 IC50 = 11220.18 nM T68251 CWEG57 155545190 IC50 = 3 nM T68251 CP6W3Q 155545205 IC50 > 10000 nM T68251 CLWS20 155545852 IC50 = 47863.01 nM T68251 COH0W2 155546374 IC50 = 492 nM T68251 CLT8Z2 155546617 IC50 = 2.38 nM T68251 C3FRY8 155547834 IC50 = 0.096 nM T68251 C1FP0M 155548067 IC50 = 32 nM T68251 C9AOK6 155550135 IC50 = 3000 nM T68251 C9ZUH8 155553520 IC50 = 6200 nM T68251 CPQ84I 155553728 IC50 > 10000 nM T68251 CM7C1P 155555245 IC50 = 16240 nM T68251 CS62RN 155556052 IC50 = 13803.84 nM T68251 C94NQE 155556307 IC50 > 10000 nM T68251 C9FC1W 155557598 IC50 = 3200 nM T68251 CJHM29 155557941 IC50 = 8310 nM T68251 CD3M6P 155558654 IC50 = 16870 nM T68251 CPDF57 155558916 IC50 = 57543.99 nM T68251 CG2DI6 155560100 IC50 = 8800 nM T68251 CQJ07L 155561559 IC50 = 8800 nM T68251 C3BA9L 155561798 IC50 = 5 nM T68251 CH40UO 155562232 IC50 = 4.1 nM T68251 C6SAE0 155562336 IC50 = 8.9 nM T68251 CD18KU 155563750 IC50 = 7600 nM T68251 CM0LN1 155563771 IC50 = 810 nM T68251 CQ4WE0 155563852 IC50 = 28183.83 nM T68251 C29SMF 155565303 IC50 > 10000 nM T68251 C51ZMC 155565586 IC50 = 700 nM T68251 CZ0WK1 155566979 IC50 = 3800 nM T68251 CP9YX2 155567218 IC50 = 2400 nM T68251 C8D5VK 155567855 IC50 = 3500 nM T68251 CHL0F3 155567858 IC50 > 10000 nM T68251 C5U9LI 155569346 IC50 = 570 nM T68251 CLT4Y6 10138589 Ki = 300 nM T68251 C5U3AO 57394286 IC50 = 23 nM T68251 C0YL9R 9975488 IC50 = 1900 nM T68251 D00RNA 44446270 IC50 = 200 nM T68251 D00TRF 44423683 IC50 = 94000 nM T68251 D01UNE 44580457 Ki = 30 nM T68251 D02ECA 448942 IC50 > 100000 nM T68251 D02EFQ 10549609 IC50 = 5 nM T68251 D02UYR 9907830 Ki = 0.3 nM T68251 D03AMR 9849669 Ki = 7 nM T68251 D04GOO 10111838 IC50 > 100000 nM T68251 D04PAW 16216218 IC50 = 60000 nM T68251 D04VPH 45376872 IC50 = 18000 nM T68251 D04WWO 9889867 Ki > 3333 nM T68251 D05BMD 44423684 IC50 = 137000 nM T68251 D05JPV 44406790 IC50 = 3070 nM T68251 D05THD 44478925 IC50 = 1300 nM T68251 D06EHW 11625778 IC50 = 35 nM T68251 D06HSC 136117931 IC50 = 65000 nM T68251 D06NDR 44423687 IC50 = 81800 nM T68251 D06ZRX 5281717 IC50 = 27600 nM T68251 D07DRT 46175162 Ki = 3.8 nM T68251 D07GEL 10344307 Ki = 1.1 nM T68251 D07MJD 44479701 IC50 = 510 nM T68251 D07VXX 16721024 IC50 = 151000 nM T68251 D08ICI 44446277 IC50 = 590 nM T68251 D08NSS 5288596 IC50 < 0.1 nM T68251 D09GIL 66160 IC50 = 50000 nM T68251 D09USO 5277466 IC50 > 100000 nM T68251 D09ZOA 25049753 IC50 = 2 nM T68251 D0A0FY 44479457 IC50 = 35000 nM T68251 D0A4TC 446504 IC50 = 3 nM T68251 D0A5MV 11581319 IC50 = 1660 nM T68251 D0B3UN 44580458 Ki = 192 nM T68251 D0D7GL 10789 IC50 = 146000 nM T68251 D0E5MB 44411812 IC50 = 792 nM T68251 D0F2HJ 45257111 IC50 = 196500 nM T68251 D0F7BE 4369084 Ki = 3000 nM T68251 D0FO2B 1923 IC50 = 130000 nM T68251 D0G0OP 44423685 IC50 = 68000 nM T68251 D0G3YZ 11391583 IC50 = 4520 nM T68251 D0H2PA 9886977 Ki = 0.5 nM T68251 D0H6CK 10160968 Ki > 3333 nM T68251 D0J0WJ 45257110 IC50 = 232500 nM T68251 D0K4TI 49292 IC50 = 1300 nM T68251 D0L4EO 11609208 IC50 = 440 nM T68251 D0L6ND 10089677 IC50 = 1.7 ug.mL-1 T68251 D0N8YA 159596 IC50 = 15000 nM T68251 D0NP8A 10370504 IC50 = 1790 nM T68251 D0NV9C 22004198 IC50 = 40 nM T68251 D0P2TS 9818682 IC50 > 60000 nM T68251 D0Q4TA 10044321 IC50 = 12 nM T68251 D0Q9LC 44385624 IC50 = 868 nM T68251 D0R2BO 194777 IC50 = 0.7 nM T68251 D0S9OL 10155934 IC50 = 1200 nM T68251 D0T1FR 44457233 IC50 = 4000 nM T68251 D0UI1P 46228278 IC50 = 178600 nM T68251 D0V9EN 689043 IC50 = 24.26 nM T68251 D0VI2A 44447430 IC50 = 537 nM T68251 D0W2UK 6914621 Ki = 2050 nM T68251 D0W3ME 4369080 Ki = 3000 nM T68251 D0XK7G 10445302 IC50 = 32 nM T68251 D0Y1XM 44423686 IC50 = 33700 nM T68251 D0Y5IQ 44255320 IC50 = 5000 nM T68251 D0Y7NV 2220392 IC50 = 898 nM T68251 D0Z4LO 9832179 IC50 = 23 nM T68251 D0Z4NU 46228282 IC50 = 285900 nM T72319 CV39DH 1072048 Ki = 33100 nM T72319 C64ZSL 43430547 IC50 > 30000 nM T72319 CQ4P5B 44755448 IC50 > 30000 nM T72319 C3NE8O 46931242 IC50 > 30000 nM T72319 C6O8RT 55872720 IC50 > 30000 nM T72319 C2P7SD 56577044 IC50 > 10000 nM T72319 CXY3E4 57720618 IC50 > 30000 nM T72319 CY9Z8F 60735522 IC50 > 30000 nM T72319 CB0SA4 61041645 IC50 > 30000 nM T72319 CT9M2C 61041646 IC50 > 30000 nM T72319 C3I5DM 61041804 IC50 > 30000 nM T72319 C84MGB 61242835 IC50 > 30000 nM T72319 C0Y6KO 62947261 IC50 > 30000 nM T72319 C8XEI4 63259457 IC50 > 30000 nM T72319 C0WX5O 70679311 IC50 > 30000 nM T72319 CEW3R6 71598546 IC50 > 30000 nM T72319 CUD65X 73333125 IC50 > 10000 nM T72319 CHQ18I 73333126 IC50 > 10000 nM T72319 C9UDN1 73333127 IC50 > 10000 nM T72319 C9K1NV 73333128 IC50 > 10000 nM T72319 C4UE6G 73333129 IC50 > 10000 nM T72319 CV2SJ4 73333225 IC50 > 10000 nM T72319 CF8HO3 73333226 IC50 > 10000 nM T72319 CVH9F0 73333227 IC50 > 10000 nM T72319 C4PYG2 73333229 IC50 > 10000 nM T72319 CBJC52 73333322 IC50 > 10000 nM T72319 CVEN67 73334066 IC50 > 10000 nM T72319 CYL3M7 73334067 IC50 > 10000 nM T72319 C6T7YX 73334068 IC50 > 10000 nM T72319 C70XCT 73334069 IC50 > 10000 nM T72319 C8QWP1 73334070 IC50 > 10000 nM T72319 CR98DL 73334157 IC50 > 10000 nM T72319 CJD9C1 73334158 IC50 > 10000 nM T72319 CLRM71 73334159 IC50 > 10000 nM T72319 C43NER 73334160 IC50 > 10000 nM T72319 CD2HX4 73334161 IC50 > 10000 nM T72319 CC89FN 73334162 IC50 > 10000 nM T72319 COV3R1 73334262 IC50 > 10000 nM T72319 CZD0N1 73334263 IC50 > 10000 nM T72319 CU3KG0 73334264 IC50 > 10000 nM T72319 CMLV27 73334265 IC50 > 10000 nM T72319 CD0VK7 73334266 IC50 > 10000 nM T72319 C1SGJ3 73334267 IC50 > 10000 nM T72319 C3PYF5 73334361 IC50 > 10000 nM T72319 C8H9JF 73334363 IC50 > 10000 nM T72319 C8XE1J 73334364 IC50 > 10000 nM T72319 CN40ZI 73334365 IC50 > 10000 nM T72319 CF9GA5 73334366 IC50 > 10000 nM T72319 C69WLM 73334479 IC50 > 10000 nM T72319 CG32QB 73334480 IC50 > 10000 nM T72319 CVE0S2 73334481 IC50 > 10000 nM T72319 C2S8XN 73334482 IC50 > 10000 nM T72319 CXJP87 73334483 IC50 > 10000 nM T72319 C57KSE 73334484 IC50 > 10000 nM T72319 CAQ18T 73334592 IC50 > 10000 nM T72319 CA67YG 73334593 IC50 > 10000 nM T72319 CNS84D 73334594 IC50 > 10000 nM T72319 C93HWE 73334595 IC50 > 10000 nM T72319 C87UBE 73334596 IC50 > 10000 nM T72319 CKSY83 73334696 IC50 > 10000 nM T72319 C36QHM 73334697 IC50 > 10000 nM T72319 CF63HU 73334698 IC50 > 10000 nM T72319 CQBX27 73334699 IC50 > 10000 nM T72319 C0OW1V 73334700 IC50 > 10000 nM T72319 C2VFJ9 73349256 IC50 > 30000 nM T72319 CG80NF 73349257 IC50 > 10000 nM T72319 COY1J2 73349259 IC50 > 10000 nM T72319 CNO9Z5 73350843 IC50 > 10000 nM T72319 C8U0ZX 73352326 IC50 > 10000 nM T72319 CRZ62F 73355036 IC50 = 8100 nM T72319 CD26ZM 73386663 IC50 = 73000 nM T72319 C2OXQ5 76314887 IC50 > 30000 nM T72319 C3X7EW 76314888 IC50 > 30000 nM T72319 C1YKN5 76314889 IC50 > 30000 nM T72319 C4E1BN 76318504 IC50 > 30000 nM T72319 CF76CT 76318505 IC50 > 30000 nM T72319 CLVA91 76318506 IC50 > 30000 nM T72319 C9LNK4 76318507 IC50 > 30000 nM T72319 CL87KC 76318508 IC50 > 30000 nM T72319 CET23F 76318509 IC50 > 30000 nM T72319 C01JLF 76322168 IC50 > 30000 nM T72319 C2SEM0 76322169 IC50 > 30000 nM T72319 CRH48X 76322170 IC50 > 30000 nM T72319 C5CZV2 76325789 IC50 > 30000 nM T72319 CS6GL0 76333019 IC50 > 30000 nM T72319 C7IUX5 76333020 IC50 > 30000 nM T72319 CZC8W2 76336632 IC50 > 30000 nM T72319 CYQ0B9 76336633 IC50 > 30000 nM T72319 CK2N0L 76336634 IC50 > 30000 nM T72319 CS4W5I 76336635 IC50 > 30000 nM T72319 CM6H9O 76336636 IC50 > 30000 nM T72319 CL8E1A 83748040 IC50 > 30000 nM T72319 CK5MX8 90655573 IC50 = 11000 nM T72319 C0S3XK 90655574 IC50 = 6800 nM T72319 CC50PO 90655575 IC50 = 5700 nM T72319 CA07UL 90655576 IC50 = 67000 nM T72319 CSUT18 90655577 IC50 = 23000 nM T72319 CD43OR 90655578 IC50 = 62000 nM T72319 C2A3RQ 90655579 IC50 = 35000 nM T72319 CEOP54 90655580 IC50 = 10100 nM T72319 CAM67V 90655581 IC50 = 10300 nM T72319 CLR17Q 90655582 IC50 = 13000 nM T72319 C28HZW 90655583 IC50 = 11000 nM T72319 CA1Y5I 90655584 IC50 = 21000 nM T72319 CQY83C 90655585 IC50 = 11200 nM T72319 CQTF13 90655586 IC50 = 6000 nM T72319 C83EFC 90655587 IC50 = 8800 nM T72319 C25ZNR 90655588 IC50 = 39000 nM T72319 C0GIC4 90655589 IC50 = 120000 nM T72319 CR6VS0 90655590 IC50 = 53000 nM T72319 C6KU2N 90655591 IC50 > 500000 nM T72319 C65HLO 90655592 IC50 = 9000 nM T72319 C4ACU9 90655593 IC50 = 79000 nM T72319 C74MKT 90655594 IC50 = 560000 nM T72319 CM21PY 90655595 IC50 > 250000 nM T72319 C78GYV 90655596 IC50 > 500000 nM T72319 C86DBC 90655597 IC50 > 250000 nM T72319 C9QU1T 90655598 IC50 > 250000 nM T72319 CWXY79 90655599 IC50 = 35000 nM T72319 C8M3HN 90655600 IC50 = 102000 nM T72319 C1MDL6 90655601 IC50 = 26000 nM T72319 C1MDK2 90655602 IC50 = 23000 nM T72319 CCD42S 90655603 IC50 = 22000 nM T72319 C7C9MF 90655604 IC50 = 105000 nM T72319 C27CIT 90655605 IC50 = 8600 nM T72319 C9PUC5 90655606 IC50 = 7800 nM T72319 CK2F6S 90655607 IC50 = 26000 nM T72319 C5T9WY 90655608 IC50 = 57000 nM T72319 C2EUX8 90655609 IC50 = 91000 nM T72319 C2A3CS 90655610 IC50 = 23000 nM T72319 C45VLK 90655611 IC50 = 89000 nM T72319 CN54XB 90655612 IC50 = 26000 nM T72319 C14LVC 90655613 IC50 = 67000 nM T72319 C64DAW 90655614 IC50 = 58000 nM T72319 C5H9VJ 90655615 IC50 = 100000 nM T72319 C9Z6BP 90655616 IC50 = 58000 nM T72319 C31VJO 90655617 IC50 > 250000 nM T72319 CAFW32 90655618 IC50 > 250000 nM T72319 CNZ4D8 90655619 IC50 = 34000 nM T72319 CY1PL8 90655620 IC50 = 53000 nM T72319 C5F6MO 90655621 IC50 > 2000000 nM T72319 C54UJD 90655622 IC50 > 2000000 nM T72319 C3OB0Z 90655623 IC50 = 4600 nM T72319 CW2ND5 90655624 IC50 = 6200 nM T72319 C87RLM 90655625 IC50 = 6300 nM T72319 C05HED 90655626 IC50 = 6700 nM T72319 C2BM7J 90655627 IC50 > 250000 nM T72319 CM51GQ 90655628 IC50 = 8800 nM T72319 CSL98F 90655629 IC50 = 57000 nM T72319 CLT0P1 90655635 IC50 = 27000 nM T72319 CW25YP 90666882 IC50 > 30000 nM T72319 CQI7D0 90666883 IC50 > 30000 nM T72319 C72IZG 90666884 IC50 > 30000 nM T72319 CCDK35 90666885 IC50 > 30000 nM T72319 C2DCW6 90666886 IC50 > 30000 nM T72319 CXN36J 90666887 IC50 > 30000 nM T72319 CG2S0B 90666888 IC50 > 30000 nM T72319 C19VSG 90666889 IC50 > 30000 nM T72319 CBG12J 90666890 IC50 > 30000 nM T72319 C90LPT 90666891 IC50 > 30000 nM T72319 C0IOH4 90666892 IC50 > 30000 nM T72319 C1CU2X 101043861 IC50 = 37 nM T72319 C0YL6Q 102602632 IC50 = 16000 nM T72319 C4Z1BN 102602634 IC50 = 130 nM T72319 C30MVB 127034580 IC50 = 1700 nM T72319 CR72CK 127044991 Ki = 25000 nM T72319 CVT1R7 127044992 Ki = 10000 nM T72319 CFJ30Y 127044993 Ki = 16900 nM T72319 CWA1V6 127044994 Ki = 10000 nM T72319 CMY6T7 127045145 Ki = 4800 nM T72319 CW6BT0 127045602 Ki = 39300 nM T72319 C6NBV2 134130627 IC50 = 35 nM T72319 COEW21 134131637 IC50 > 60000 nM T72319 C9XOG1 134131644 IC50 > 60000 nM T72319 CUW67R 134133875 IC50 = 240 nM T72319 CA1LH4 134133965 IC50 > 60000 nM T72319 C7PCM8 134134706 IC50 > 60000 nM T72319 C3PR2V 134134858 IC50 = 3100 nM T72319 CZB51D 134137731 IC50 = 51000 nM T72319 CKI23U 134139941 IC50 > 60000 nM T72319 C1OEI2 134140369 IC50 > 60000 nM T72319 C62JBE 134141602 IC50 = 220 nM T72319 CB20QF 134142297 IC50 > 60000 nM T72319 C29JUC 134142686 IC50 = 56 nM T72319 CS69VL 134143576 IC50 = 25000 nM T72319 C3XG2N 134144118 IC50 = 81 nM T72319 CZ83CB 134144237 IC50 = 51000 nM T72319 C48DSU 134145156 IC50 > 60000 nM T72319 C5C0HU 134145218 IC50 = 32000 nM T72319 CX1QB4 134145347 IC50 = 53000 nM T72319 C5IMF8 134145736 IC50 > 60000 nM T72319 CQX43Z 134145760 IC50 = 570 nM T72319 CX71GT 134146508 IC50 = 47 nM T72319 CE0C7P 134146658 IC50 = 740 nM T72319 CJY6D2 134146764 IC50 > 60000 nM T72319 C7NBT1 134148174 IC50 = 1700 nM T72319 C02JMB 134148668 IC50 = 61 nM T72319 CTL0D2 134149263 IC50 = 1200 nM T72319 C3BD1U 134149299 IC50 = 250 nM T72319 CS73OF 134149994 IC50 = 41000 nM T72319 C1MLU3 134151077 IC50 > 60000 nM T72319 C21YGK 134151685 IC50 > 60000 nM T72319 CES73F 134152016 IC50 = 1100 nM T72319 CIZV46 134152824 IC50 > 60000 nM T72319 C38AYE 134153154 IC50 = 230 nM T72319 CD5VJ0 134153698 IC50 = 18000 nM T72319 C4C7VM 134154055 IC50 = 75 nM T72319 CPAK59 134154083 IC50 = 4400 nM T72319 C9SAU3 134154301 IC50 = 32 nM T72319 CVK52O 134155339 IC50 = 35 nM T72319 CUH81S 134156240 IC50 = 26000 nM T72319 CB3YE8 134156251 IC50 = 63 nM T72319 CQ35RF 134157076 IC50 > 60000 nM T72319 CU0Z1S 134157587 IC50 = 28000 nM T72319 CFHK68 134157612 IC50 = 2600 nM T72319 D0W9RR 57339144 IC50 > 10000 nM T97353 D01TJY 53340771 IC50 > 10 nM T97353 CS24BW 11973730 IC50 = 15 nM T97353 CG3FV0 16727128 IC50 = 214 nM T97353 CAVY89 23636144 IC50 = 102 nM T97353 C1VUH4 23636254 IC50 = 17 nM T97353 C6LR7V 23636255 IC50 = 50 nM T97353 C5MSF6 23636502 IC50 = 29 nM T97353 C8B7QE 72949858 IC50 > 5000 nM T97353 C5ALQ2 76285468 IC50 = 4 nM T97353 CQ8BX7 76310576 IC50 = 163 nM T97353 C0JKX6 76310577 IC50 = 588 nM T97353 CUAH40 76310578 IC50 = 978 nM T97353 C4EK9U 76310579 IC50 > 4000 nM T97353 COZ54T 76310580 IC50 > 1000 nM T97353 CHI2U7 76310581 IC50 > 1000 nM T97353 COI21T 76310597 IC50 = 34 nM T97353 CL3EO0 76310599 IC50 = 470 nM T97353 CA9X2E 76310600 IC50 > 4000 nM T97353 CT1AJ4 76314216 IC50 = 114 nM T97353 C90ZKU 76314217 IC50 = 233 nM T97353 CA42YR 76314218 IC50 = 731 nM T97353 CXQ41E 76314219 IC50 > 10000 nM T97353 CUHZ51 76314232 IC50 = 667 nM T97353 COQ48X 76314233 IC50 = 1297 nM T97353 C1M7ZG 76317786 IC50 = 178 nM T97353 CIQ0T7 76317787 IC50 = 745 nM T97353 C1I6HO 76317788 IC50 = 1050 nM T97353 CSA72F 76317789 IC50 > 1000 nM T97353 CC3U8I 76317804 IC50 > 1000 nM T97353 C5UPA9 76317805 IC50 = 366 nM T97353 CBR9F0 76317806 IC50 = 36 nM T97353 CV23LI 76317807 IC50 > 5000 nM T97353 C0O4QY 76321498 IC50 = 101 nM T97353 CG7H4W 76321513 IC50 = 792 nM T97353 C1BQF4 76321514 IC50 = 38 nM T97353 C2ZH7K 76321515 IC50 = 497 nM T97353 CS9W7I 76321516 IC50 = 909 nM T97353 C7HC0P 76321517 IC50 > 4000 nM T97353 C8QH1P 76321518 IC50 = 731 nM T97353 CI9T5J 76325099 IC50 = 142 nM T97353 C2C6EW 76325100 IC50 > 4000 nM T97353 CSVC17 76325118 IC50 > 4000 nM T97353 CMH79B 76325119 IC50 = 12 nM T97353 C1HJO0 76325120 IC50 = 869 nM T97353 CCN7M6 76328682 IC50 = 1900 nM T97353 CP7AC0 76328683 IC50 > 5000 nM T97353 CX3Y7N 76328684 IC50 = 270 nM T97353 CZM19H 76332361 IC50 = 134 nM T97353 C18OJH 76332362 IC50 = 176 nM T97353 CA1LM2 76335971 IC50 = 106 nM T97353 C4I5DV 76335989 IC50 > 1000 nM T97353 CVI67F 90665342 EC50 = 2000 nM T19567 C3MA9U 342139 Ki = 3200 nM T19567 CDUE24 778225 IC50 < 200 nM T19567 CL16MS 822778 IC50 = 1000 nM T19567 CDX3Q5 5289024 Ki = 10 nM T19567 C7W8IX 5486943 Ki = 46 nM T19567 C3X1UJ 11507040 Ki = 600 nM T19567 C8N6MC 24808481 Ki = 420 nM T19567 C75WCL 52949691 Ki = 700 nM T19567 C54CBK 54585170 Ki = 5900 nM T19567 CTL94E 57520838 Ki = 9.4 nM T19567 CJQ9O0 57520839 Ki = 11 nM T19567 C8S9PM 57520840 Ki > 3000 nM T19567 C9G2HN 57520841 Ki = 50 nM T19567 C3N4MF 57520842 Ki = 29 nM T19567 CU4NZ2 57520938 Ki = 41 nM T19567 CD0M8V 57520940 Ki = 14 nM T19567 CCS1L3 57520941 Ki = 0.53 nM T19567 CEL56T 57520942 Ki = 20 nM T19567 CM6RX9 57520943 Ki = 9 nM T19567 C9Q4XE 57520944 Ki = 180 nM T19567 C1Z0LC 57520945 Ki = 1200 nM T19567 CE09OR 57520946 Ki = 200 nM T19567 C3Z6AE 57521037 Ki = 14 nM T19567 C6XB7H 57521039 Ki = 2.4 nM T19567 CXN9G4 57521040 Ki = 74 nM T19567 C9RU7B 57521041 Ki = 760 nM T19567 CC6UT9 57521043 Ki = 26 nM T19567 C78HYG 57521133 Ki = 0.36 nM T19567 C42KWH 57521134 Ki = 5.3 nM T19567 C9DFB0 57521135 Ki > 3000 nM T19567 C6SZ1P 57521138 Ki = 50 nM T19567 CR23AT 57521139 Ki = 58 nM T19567 CCQM76 59153288 Ki = 5.5 nM T19567 C4K2LU 59153299 Ki = 5.6 nM T19567 CK76DI 60202405 Ki = 2.8 nM T19567 C2LBW7 66551925 Ki = 190 nM T19567 C9CZS3 67205978 Ki = 70 nM T19567 C10MDK 69082696 Ki = 13 nM T19567 C39VMJ 69082892 Ki = 3.3 nM T19567 CYH83A 69083992 Ki = 1800 nM T19567 CT1PN0 69084444 Ki = 1700 nM T19567 CPV2D7 69085518 Ki = 960 nM T19567 CBZ82I 69085541 Ki = 72 nM T19567 CY2W3Z 69085646 Ki > 3000 nM T19567 C6BE5X 71271461 Ki = 270 nM T19567 C74PAB 86223063 Ki = 2200 nM T19567 CL0ZX5 86223064 Ki > 100000 nM T19567 CPT0J9 86275056 IC50 < 200 nM T19567 CIOU35 86275306 IC50 = 1000 nM T19567 CT4E5W 102436701 Ki = 4.1 nM T19567 C53VJW 135301646 IC50 = 3.715 nM T19567 C26OPR 135301656 IC50 = 147.91 nM T19567 CZVS32 135301671 IC50 = 3.89 nM T19567 CZJV94 135301685 IC50 = 18.2 nM T19567 CS4UK6 135301687 IC50 = 181.97 nM T19567 C9LA1K 135301762 IC50 = 20.42 nM T19567 CVW5G9 135301817 IC50 = 77.62 nM T19567 CG93EF 135301914 IC50 = 6.026 nM T19567 CGL0U2 135301919 IC50 = 13.18 nM T19567 C94GAU 135301927 IC50 = 2630.27 nM T19567 CY4MV6 135566354 Ki = 0.41 nM T19567 C4OVP2 136416802 Ki = 44 nM T19567 C7ZCT8 136416815 Ki = 69 nM T19567 C1OA7D 136416820 Ki = 0.55 nM T19567 C50OXS 136416829 Ki = 23 nM T19567 CX54DV 136416830 Ki = 28 nM T19567 CH94UL 136416849 Ki = 7.9 nM T19567 C9L0UB 136416923 Ki = 3 nM T19567 C0QWG9 142408858 IC50 = 10.23 nM T19567 CLZ91U 145971636 Ki > 200000 nM T19567 C4YPL9 145972068 Ki = 3460 nM T19567 CZVU97 155511644 Ki = 800 nM T19567 CMI8N3 155513321 Ki = 1600 nM T19567 C2CI4A 155514380 Ki = 600 nM T19567 CJ45PR 155520478 Ki = 2000 nM T19567 C95LZD 155522194 Ki = 700 nM T19567 CA35VB 155524076 Ki = 2100 nM T19567 C2QA1Z 155525301 Ki = 3200 nM T19567 C1E0UF 155535661 Ki = 3800 nM T19567 C2DI7E 155536657 IC50 = 3700 nM T19567 C3K1BZ 155537205 Ki = 15900 nM T19567 C9F2JN 155538608 Ki = 35 nM T19567 C5T9KE 155542416 Ki > 3000 nM T19567 C08TBV 155543421 IC50 = 223.87 nM T19567 C9S4MT 155549437 Ki = 1200 nM T19567 CAM36F 155550472 Ki = 3500 nM T19567 C3XE9Y 155554199 Ki = 900 nM T19567 C3WT2Q 155556441 Ki > 3000 nM T19567 C3PHB1 155557026 Ki = 2200 nM T19567 C3FA0E 155558092 Ki = 6700 nM T19567 C2I8VX 155559220 Ki = 8300 nM T19567 CUH07S 155560032 IC50 = 25000 nM T19567 CC5FE7 155564581 Ki > 3000 nM T19567 CB1V8A 155564612 Ki > 3000 nM T84621 D02STN 132971 IC50 = 1608 nM T84621 D02YPG 667484 IC50 = 0.5 nM T84621 D07ABV 468595 IC50 = 310 nM T84621 D09LNI 3365 IC50 = 30000 nM T84621 D0C1WH 3902 IC50 = 2620 nM T84621 D0Q9JT 4174 IC50 = 14.6 nM T84621 D0ZX1P 59693 IC50 = 6.3 nM T84621 D03AJU 44139752 IC50 = 2.5 nM T84621 D0D3PF 6918191 IC50 = 95000 nM T84621 D0SX7F 60876 Ki = 35 nM T84621 C9LCD8 3823 IC50 = 127 nM T84621 CFO8Y3 83332 IC50 = 24800 nM T84621 C78IXN 563347 IC50 = 246 nM T84621 CNG05O 571156 IC50 = 779 nM T84621 C5NT4U 583968 IC50 = 24 nM T84621 C1Y5HM 603115 IC50 = 16700 nM T84621 C8HZL4 618231 IC50 = 3 nM T84621 C7XD4N 706178 IC50 = 10200 nM T84621 CJ4FE1 853038 IC50 = 635 nM T84621 CI16RF 867617 IC50 = 500 nM T84621 CC29WP 886929 IC50 = 194 nM T84621 C6S1WJ 955210 IC50 > 1000 nM T84621 CB5KN2 1118253 IC50 = 14300 nM T84621 C83OBD 3021561 IC50 = 763 nM T84621 CBY4W2 3102914 IC50 > 1000 nM T84621 C1JAT6 6539761 IC50 = 715 nM T84621 CTE57C 6539762 IC50 = 1424 nM T84621 CF17BE 6539771 IC50 = 903 nM T84621 CJ7RS8 6539772 IC50 = 206 nM T84621 CQD13Z 6539787 IC50 = 143 nM T84621 CQ0HD5 6539812 IC50 = 58 nM T84621 CQ9XM0 6539813 IC50 = 26 nM T84621 CP51TH 6539814 IC50 = 96 nM T84621 CP4VI2 6540030 IC50 = 31.4 nM T84621 CR6LS8 6540031 IC50 = 3.3 nM T84621 CU3C1Y 6540034 IC50 = 6.9 nM T84621 CXEW82 6540035 IC50 = 15 nM T84621 CBKX32 6540037 IC50 = 18.7 nM T84621 C8MRI7 6540038 IC50 = 20.6 nM T84621 C8JXY1 6540039 IC50 = 11.17 nM T84621 CZK3T4 6540040 IC50 = 28.7 nM T84621 CDS26H 6540041 IC50 = 19.5 nM T84621 CX38PV 9927427 IC50 = 2 nM T84621 C64PHS 10083522 IC50 = 75000 nM T84621 CTH96I 10584844 IC50 = 5 nM T84621 CA13SW 10711620 IC50 = 79 nM T84621 CZW6V4 10828130 IC50 = 13.4 nM T84621 C6G3JV 11032034 IC50 = 47.86 nM T84621 C1TP7W 11232831 IC50 = 72 nM T84621 CN4T0K 11544009 IC50 = 4898 nM T84621 C9IJ3T 11594132 IC50 = 10505 nM T84621 CW2B3A 11738647 IC50 = 933 nM T84621 C27WEU 12229396 IC50 = 32 nM T84621 CCU19N 13045366 IC50 = 61 nM T84621 C4ELY3 13276694 IC50 = 2848 nM T84621 C1F5IT 13688212 IC50 = 40 nM T84621 C8WU6R 14424120 IC50 = 663 nM T84621 C8LSJ6 15182477 IC50 = 76000 nM T84621 CQ03PZ 16654684 IC50 = 816 nM T84621 CY0RV3 18668566 IC50 = 15 nM T84621 CRDM03 18679298 IC50 = 48 nM T84621 CN8IQ3 18785133 IC50 = 30.9 nM T84621 C1R2FU 22406650 IC50 = 253 nM T84621 C6D2NZ 24692916 IC50 = 1000 nM T84621 C07XJP 24696760 IC50 = 7500 nM T84621 CW3C5U 24896569 IC50 = 4329 nM T84621 C29WQM 25033651 IC50 = 291 nM T84621 C1VPF8 25033652 IC50 = 3109 nM T84621 C9Q8ZK 25033657 IC50 > 20000 nM T84621 CWIC10 25033659 IC50 > 10000 nM T84621 CAI47X 25033725 IC50 > 5000 nM T84621 C1XW6O 25033727 IC50 = 2135 nM T84621 CW5A1U 25033730 IC50 = 1159 nM T84621 CV49HP 25033731 IC50 = 686 nM T84621 C86AIT 25033734 IC50 > 10000 nM T84621 CEJ89P 25033804 IC50 = 2748 nM T84621 C3UF1V 25033806 IC50 = 1076 nM T84621 CF46OB 25033808 IC50 > 20000 nM T84621 CBI59C 25033810 IC50 = 1370 nM T84621 CV19DG 25034278 IC50 = 461 nM T84621 CEP93C 25034345 IC50 = 100 nM T84621 CSX16E 25034347 IC50 = 15 nM T84621 CXDF80 25034348 IC50 = 255 nM T84621 C56WJS 25034349 IC50 = 199 nM T84621 CGD93B 25034350 IC50 = 614 nM T84621 CK3L1J 25034351 IC50 = 1760 nM T84621 C9MF8O 25034425 IC50 = 99 nM T84621 CW7V9I 25034428 IC50 = 64 nM T84621 CH6U1E 25034429 IC50 = 248 nM T84621 CLP17I 25034432 IC50 = 875 nM T84621 CTB95M 25034489 IC50 = 41557 nM T84621 CBLS47 25034490 IC50 = 37796 nM T84621 CW82MN 25034491 IC50 = 31 nM T84621 CJ8M0E 25034492 IC50 = 435 nM T84621 COSJ63 25034493 IC50 = 10 nM T84621 C7KAR1 25034657 IC50 > 10000 nM T84621 C0MEI5 25129119 IC50 = 1956 nM T84621 C2QU1N 25129120 IC50 = 3559 nM T84621 C2FE6G 25129122 IC50 = 2452 nM T84621 CJ48LA 25129123 IC50 = 785 nM T84621 CX4GM7 25129462 IC50 = 24003 nM T84621 C9IFV2 25129463 IC50 = 19816 nM T84621 C6D8UQ 25129464 IC50 = 11307 nM T84621 CJCE15 25130854 IC50 = 1811 nM T84621 C9AS7H 25131165 IC50 = 2936 nM T84621 C9G8MJ 25131494 IC50 = 735 nM T84621 CA7OP2 25131495 IC50 = 9639 nM T84621 CZX08M 25142015 Ki = 15 nM T84621 C1WM2B 25147691 IC50 = 6.9 nM T84621 CYT15G 25180102 IC50 = 5970 nM T84621 CGX76Y 25180105 IC50 = 4371 nM T84621 CMU54R 25180107 IC50 = 290 nM T84621 C0XHA2 25180109 IC50 = 742 nM T84621 C9LQJ6 25180110 IC50 = 5177 nM T84621 CHJ2S3 25180298 IC50 = 339 nM T84621 C1HGB6 25180299 IC50 = 1671 nM T84621 C90UKD 25180304 IC50 = 1145 nM T84621 CPQ6A9 25180305 IC50 = 745 nM T84621 C6ZE9H 25180500 IC50 = 191 nM T84621 C6FN2Z 25180502 IC50 = 5402 nM T84621 C9DB1G 25180503 IC50 = 87 nM T84621 CIZ82U 25180504 IC50 = 769 nM T84621 CJS97E 30507078 IC50 = 5920 nM T84621 C70VMZ 44203017 IC50 = 1987 nM T84621 CT3XM4 44206480 IC50 = 116 nM T84621 C9UWB5 44206481 IC50 = 57 nM T84621 CDTS58 44387709 IC50 = 12.3 nM T84621 CT4L0R 44455927 IC50 = 19 nM T84621 C69QUY 44456068 IC50 > 1000 nM T84621 CM8BT1 44456104 IC50 = 110 nM T84621 C68FJH 44456188 IC50 = 167 nM T84621 CP50NM 44456189 IC50 = 329 nM T84621 CVR70K 44456190 IC50 = 782 nM T84621 C9JCL1 44456223 IC50 = 213 nM T84621 C6BE0T 44456226 IC50 = 107 nM T84621 CO4PI7 44479388 IC50 = 715 nM T84621 C1K6QY 44479389 IC50 = 2296 nM T84621 CLPH49 44479390 IC50 = 247 nM T84621 C2EM5N 44479391 IC50 = 13 nM T84621 CNTI30 44479392 IC50 = 545 nM T84621 C40IPE 44479393 IC50 = 34 nM T84621 C8JHS9 44479641 IC50 = 333 nM T84621 C2P4XT 44479643 IC50 = 158 nM T84621 CWP4Y8 44479644 IC50 = 141 nM T84621 C81QJE 44479645 IC50 = 1288 nM T84621 CO8T3N 44479646 IC50 = 2077 nM T84621 C4YN0S 44479648 IC50 = 28546 nM T84621 CF12OV 44479882 IC50 = 58 nM T84621 CCN58W 44479883 IC50 = 103 nM T84621 C7GV6X 44479884 IC50 = 17 nM T84621 CH8RO1 44479885 IC50 = 40 nM T84621 CES96D 44479886 IC50 = 490 nM T84621 CH02ZN 44480128 IC50 = 21 nM T84621 C1LSH2 44480129 IC50 = 1374 nM T84621 C3UQS0 44480130 IC50 = 43 nM T84621 C4KG5O 44480131 IC50 = 4646 nM T84621 COI7E8 44480132 IC50 = 496 nM T84621 C9KS5O 44480133 IC50 = 2058 nM T84621 CLMI41 44480134 IC50 = 128 nM T84621 CYH9A6 44480385 IC50 = 1312 nM T84621 C9V8CH 44480386 IC50 = 28 nM T84621 CL8KQ3 44480387 IC50 = 54 nM T84621 CT50NZ 44480388 IC50 = 796 nM T84621 CKO4N3 44480389 IC50 = 1692 nM T84621 CT3MO9 44480390 IC50 = 15 nM T84621 CN7LT2 44482245 IC50 = 776 nM T84621 CO63LK 44569291 IC50 = 152 nM T84621 CW06BV 45103704 IC50 = 104 nM T84621 C9Z4YB 45103705 IC50 = 123 nM T84621 CB2FC9 45103804 IC50 = 112.2 nM T84621 C4Q2FU 45103806 IC50 = 43.65 nM T84621 CQF56Z 45103807 IC50 = 12.02 nM T84621 C0RY2G 46233602 IC50 = 213 nM T84621 CUV83E 46854605 IC50 = 3100 nM T84621 CIA08B 46854608 IC50 = 37470 nM T84621 CWJ3F1 46854758 IC50 = 7300 nM T84621 CKRQ67 46854759 IC50 = 7180 nM T84621 CZ1YJ0 46854760 IC50 = 5060 nM T84621 CIC9S5 49799473 IC50 = 2000 nM T84621 C3Q6AS 49862488 IC50 = 26.1 nM T84621 CM43HV 49862547 IC50 = 50.2 nM T84621 CFDH59 49862548 IC50 = 103 nM T84621 CNIA98 49862549 IC50 = 544 nM T84621 CKY2J9 49862550 IC50 = 566 nM T84621 C0N4RT 49862551 IC50 = 930 nM T84621 CLI23H 49862552 IC50 = 122 nM T84621 CGU86D 49862599 IC50 = 55.7 nM T84621 CY8WD5 49862600 IC50 = 119 nM T84621 CS4IP9 49862601 IC50 = 76 nM T84621 C63XUS 49862602 IC50 = 204 nM T84621 C6O7JQ 49862603 IC50 = 471 nM T84621 C8G7FR 49862604 IC50 = 340 nM T84621 CP5D8Q 49862650 IC50 = 20.6 nM T84621 C6X0JA 49862651 IC50 = 222 nM T84621 C7BTK9 49862652 IC50 = 245 nM T84621 C79MQZ 49862653 IC50 = 234 nM T84621 CL8DR6 49862654 IC50 = 182 nM T84621 CMXR96 51355428 IC50 = 45 nM T84621 C5KTL3 51355429 IC50 = 40 nM T84621 C4UTM8 51355430 IC50 = 31 nM T84621 CH5C9K 51355431 IC50 = 20 nM T84621 CRK2Q9 51355432 IC50 = 5 nM T84621 CF7RG5 51355433 IC50 = 20 nM T84621 C41SUK 51355703 IC50 = 100 nM T84621 CM6T7H 51355704 IC50 = 80 nM T84621 CZDA87 51355705 IC50 = 25 nM T84621 CO1V0Y 51355706 IC50 = 45 nM T84621 C2OCG3 51355707 IC50 = 50 nM T84621 CIR0L7 51356252 IC50 = 933 nM T84621 CY69GL 52450897 IC50 = 188 nM T84621 CMTX50 52936939 IC50 = 2045 nM T84621 CC7Q8A 52936940 IC50 = 183 nM T84621 CTD3M1 52936941 IC50 = 1748 nM T84621 C98MZS 52937039 IC50 = 44 nM T84621 CZ72GJ 53316510 IC50 = 46 nM T84621 CR7L6V 53317838 IC50 = 80 nM T84621 CD9JL4 53319024 IC50 = 16100 nM T84621 CJBC94 53319146 IC50 > 1000 nM T84621 CYN7S9 53319147 IC50 = 43 nM T84621 C6WXT3 53320325 IC50 = 369 nM T84621 C20LRW 53320468 IC50 = 32 nM T84621 CU80BY 53320469 IC50 > 1000 nM T84621 C1SH0Q 53321768 IC50 > 1000 nM T84621 CEA3Y9 53321769 IC50 > 1000 nM T84621 C90DZC 53322953 IC50 = 5 nM T84621 CU1V2C 53323093 IC50 = 128 nM T84621 CYU1S5 53323094 IC50 > 1000 nM T84621 CS4A9O 53324450 IC50 = 46 nM T84621 C0B7TL 53325759 IC50 = 197 nM T84621 CVG4U6 53325760 IC50 = 4 nM T84621 CO68YD 53326854 IC50 = 75 nM T84621 C4NU2F 53475401 IC50 = 42 nM T84621 CAE25J 53763992 IC50 = 500 nM T84621 C51RVD 56645155 IC50 = 2857 nM T84621 CG06MB 56645361 IC50 = 401 nM T84621 CUS9L4 56645362 IC50 = 3984 nM T84621 C4N0WL 56645363 IC50 = 100 nM T84621 CTO1X9 56645364 IC50 = 370 nM T84621 C57NSZ 56645568 IC50 = 42 nM T84621 C6PUX9 56645570 IC50 = 435 nM T84621 CTW6K2 56645571 IC50 = 258 nM T84621 CX05HC 56645572 IC50 = 723 nM T84621 CPCW12 56645777 IC50 = 374 nM T84621 C32FWC 56645967 IC50 = 251 nM T84621 CXYW61 56645969 IC50 = 334 nM T84621 C2AP7F 56646158 IC50 = 435 nM T84621 CKWB83 56646160 IC50 = 477 nM T84621 CA3VO0 56949328 IC50 > 7500 nM T84621 CH8CP7 57329709 IC50 = 246 nM T84621 CQD5B4 57329785 IC50 = 76 nM T84621 C8GUF0 57329786 IC50 = 29 nM T84621 CE4YX9 57329787 IC50 = 40 nM T84621 CRAD59 57329788 IC50 = 72 nM T84621 CH8FQ9 57329789 IC50 = 101 nM T84621 C4USR5 57329791 IC50 = 62 nM T84621 C2C5PD 57329792 IC50 = 75 nM T84621 C3D8CZ 57329793 IC50 = 16 nM T84621 CKH02M 57329866 IC50 = 61 nM T84621 C30NOK 57329940 IC50 = 33 nM T84621 C37KZO 57329941 IC50 = 28 nM T84621 CZH28K 57329942 IC50 = 12 nM T84621 CR6EH0 57329943 IC50 = 151 nM T84621 CWN9V2 57329944 IC50 = 60 nM T84621 CFLA57 57330005 IC50 = 21 nM T84621 C2JR3S 57330006 IC50 = 11 nM T84621 C1EZM8 57330007 IC50 = 124 nM T84621 C5H2LE 57330008 IC50 = 69 nM T84621 C05XKT 57330009 IC50 = 98 nM T84621 C26GFC 57330010 IC50 = 32 nM T84621 CS38WC 57330011 IC50 = 6 nM T84621 C54EUF 57330012 IC50 = 1122 nM T84621 C4MN9B 57330078 IC50 = 1711 nM T84621 C5K3VT 57330079 IC50 = 240 nM T84621 C3LVG9 57330084 IC50 = 610 nM T84621 CMNH08 57330085 IC50 = 8 nM T84621 CY58ZD 57330086 IC50 = 2 nM T84621 C7OK1X 57775654 IC50 = 149 nM T84621 CB6RN7 58255346 IC50 = 50 nM T84621 CFXY47 58255349 IC50 = 29 nM T84621 C34JIZ 58255359 IC50 = 224 nM T84621 C7ZH6D 58255361 IC50 = 3.4 nM T84621 C2TUJ7 58255382 IC50 = 2.2 nM T84621 CMBV34 58255389 IC50 = 40 nM T84621 C3DPC0 58255407 IC50 = 40 nM T84621 C9DK1X 58255415 IC50 = 3737 nM T84621 CQEW75 58255430 IC50 = 144 nM T84621 CTI0D7 58255435 IC50 = 5399 nM T84621 C7L1NK 58255436 IC50 = 27 nM T84621 CRQ70M 58255438 IC50 = 1.4 nM T84621 C72VNQ 58255447 IC50 = 6.5 nM T84621 CLQ65O 58255479 IC50 = 347 nM T84621 CP6RA9 58255482 IC50 = 11940 nM T84621 C6DHG3 58255496 IC50 = 70 nM T84621 CAJ17Z 58255506 IC50 = 13 nM T84621 C7AX1R 58255531 IC50 = 110 nM T84621 CJX70M 58255566 IC50 = 745 nM T84621 C64JZC 58255572 IC50 = 438 nM T84621 CW71EO 58255581 IC50 = 2487 nM T84621 CYD9N5 58255637 IC50 = 20 nM T84621 CB7N8A 60195126 IC50 = 19 nM T84621 CX4N0I 62707515 IC50 = 790 nM T84621 CH3QU4 62918897 IC50 = 971 nM T84621 CE6L7O 65040275 IC50 > 10000 nM T84621 C0G3LA 66559847 IC50 = 1098 nM T84621 C4RSI6 66559935 IC50 = 1077 nM T84621 CDX7I8 66559936 IC50 = 1167 nM T84621 CF9EQ5 66559939 IC50 = 1422 nM T84621 CQN6D3 66559940 IC50 = 16170 nM T84621 CN4H8G 66559941 IC50 = 4087 nM T84621 CTP6Q4 66559942 IC50 = 4589 nM T84621 C9EGW2 66575742 IC50 = 3570 nM T84621 CMXA10 66575743 IC50 = 1770 nM T84621 CKWB91 66575744 IC50 = 110 nM T84621 C7I3MW 66575745 IC50 = 16990 nM T84621 CPN17S 66575746 IC50 = 12620 nM T84621 CG0ZA7 66575747 IC50 = 16100 nM T84621 C6HF0U 66575748 IC50 = 7900 nM T84621 CEW4O6 66575816 IC50 = 17296 nM T84621 CDI93T 66575817 IC50 = 428 nM T84621 C6B7PN 66576767 IC50 = 407 nM T84621 CYHS25 66576769 IC50 = 1501 nM T84621 CBP6I7 66576773 IC50 = 2198 nM T84621 CM6U5S 66576848 IC50 > 30000 nM T84621 CNB21T 66576849 IC50 > 10000 nM T84621 C2PFB6 66576850 IC50 > 10000 nM T84621 CDU8R7 66576852 IC50 = 6930 nM T84621 C4NYB0 66576930 IC50 = 1810 nM T84621 C3LP5H 66576931 IC50 = 3910 nM T84621 CE03WG 66576932 IC50 = 6970 nM T84621 CVZ4E0 66692998 IC50 > 10000 nM T84621 C1RLT0 67199421 IC50 = 3451 nM T84621 CC34QF 67509960 IC50 = 21 nM T84621 CQL7H6 67510362 IC50 = 167 nM T84621 CN9VU2 67510431 IC50 = 320 nM T84621 C40FEA 67511528 IC50 = 362 nM T84621 C2MH1G 67515607 IC50 = 126 nM T84621 CC4A7Z 67515696 IC50 = 106 nM T84621 CE27NZ 67515801 IC50 = 782 nM T84621 CZCW84 67515869 IC50 = 362 nM T84621 CKJN74 67515874 IC50 = 409 nM T84621 CW20PM 67516106 IC50 = 502 nM T84621 C14VNF 67516160 IC50 = 1000 nM T84621 CL0XQ7 67516179 IC50 = 971 nM T84621 CM7Z1T 67516370 IC50 = 95 nM T84621 CK1LB2 67516475 IC50 = 542 nM T84621 C5VM6T 67516855 IC50 = 139 nM T84621 CQ0NP7 68053462 IC50 > 10000 nM T84621 CV72CY 68053552 IC50 = 1980 nM T84621 CVF40X 68053622 IC50 = 1831 nM T84621 CG0T8B 68053623 IC50 = 2101 nM T84621 CU76KO 68053624 IC50 > 8333 nM T84621 CYZK18 68053631 IC50 > 8333 nM T84621 CSI12Z 68053632 IC50 > 10000 nM T84621 C0N3IK 68053729 IC50 = 17.7 nM T84621 C19JSA 68053730 IC50 = 250 nM T84621 C5N2MQ 68053837 IC50 = 677 nM T84621 CCJT39 68053838 IC50 = 3923 nM T84621 CF32HJ 70680985 IC50 = 500 nM T84621 CPB63L 70680997 IC50 = 73 nM T84621 CE78SM 70683110 IC50 = 168 nM T84621 CM6LN8 70683111 IC50 = 246 nM T84621 CK0DY6 70683112 IC50 = 611 nM T84621 C9E4ZQ 70685192 IC50 = 269 nM T84621 CW5F3G 70691516 IC50 = 500 nM T84621 C1VMF2 70977969 IC50 = 29540 nM T84621 C70TUP 71455138 IC50 = 139 nM T84621 CFG4L5 71456934 IC50 = 44 nM T84621 CI16NC 71520311 IC50 = 1336 nM T84621 CE9A6B 71520312 IC50 > 5000 nM T84621 C03VKJ 71520313 IC50 = 750 nM T84621 C5J7DI 71520314 IC50 = 16 nM T84621 CE0N5C 71520315 IC50 = 41 nM T84621 C4Z6YP 71520316 IC50 = 1230 nM T84621 CC8Z6L 71520431 IC50 = 4 nM T84621 C1DK9P 71520432 IC50 = 140 nM T84621 C9NOQ1 71521632 IC50 = 68 nM T84621 C0OTA2 71521716 IC50 = 2270 nM T84621 CVLE07 71521717 IC50 = 1220 nM T84621 CJKX84 71521718 IC50 = 36 nM T84621 CZ5P9U 71521719 IC50 = 78 nM T84621 C1YCB0 71521720 IC50 = 1420 nM T84621 CE57PM 71521721 IC50 > 5000 nM T84621 C0O2SA 71521798 IC50 = 276 nM T84621 CMEC10 71521799 IC50 = 2539 nM T84621 CR9O5T 71521800 IC50 = 1688 nM T84621 C0JBI3 71521801 IC50 = 532 nM T84621 CE7Z4I 71521802 IC50 = 88 nM T84621 CW2AG4 71521803 IC50 = 646 nM T84621 C6ID7K 71521804 IC50 = 92 nM T84621 CO5BE7 71535395 IC50 = 280 nM T84621 CCF8Z7 71535398 IC50 = 530 nM T84621 CC16AO 71535399 IC50 = 590 nM T84621 CPZ5S8 71535400 IC50 = 100 nM T84621 CI4W5N 71535682 IC50 = 490 nM T84621 CCRS95 71535683 IC50 = 1800 nM T84621 C58SMB 71574941 IC50 = 0.5 nM T84621 CC09FQ 71574942 IC50 = 19.2 nM T84621 CA2T5L 71574943 IC50 = 156.3 nM T84621 C9MFZ7 71574944 IC50 = 80.1 nM T84621 CW73OE 71574945 IC50 = 25.4 nM T84621 C70NHJ 71574946 IC50 = 92.5 nM T84621 CLH83S 71574947 IC50 = 24.4 nM T84621 CF71AB 71575030 IC50 = 13.1 nM T84621 CCG1S5 71575031 IC50 = 5.5 nM T84621 CH9WE7 71575032 IC50 = 268.4 nM T84621 CO4ZQ7 71575033 IC50 = 415.8 nM T84621 CT86GV 71575034 IC50 = 785.3 nM T84621 CKPV51 71621803 IC50 > 100000 nM T84621 CG09JH 71716351 IC50 = 72 nM T84621 C56LUJ 71716957 IC50 = 219 nM T84621 CJE01S 71745100 IC50 = 4520 nM T84621 CX0WV5 71817943 IC50 = 235 nM T84621 CN1LU6 71817944 IC50 = 1609 nM T84621 CGV4U3 71817945 IC50 = 1159 nM T84621 CJ4L5G 71818086 IC50 = 2935 nM T84621 COXA51 71818087 IC50 = 224 nM T84621 CP1A3M 71818088 IC50 = 1415 nM T84621 CPJ42T 71818089 IC50 = 450 nM T84621 CAP03I 71818090 IC50 = 447 nM T84621 CO23PK 71818091 IC50 = 245 nM T84621 CL4X6A 71818092 IC50 = 7099 nM T84621 CL8GK5 71818093 IC50 = 2824 nM T84621 C4ZVG0 71818094 IC50 = 362 nM T84621 CH2GR0 71818232 IC50 = 238 nM T84621 C0VGQ9 71818233 IC50 = 12286 nM T84621 C5QRF2 71818234 IC50 = 2426 nM T84621 CCG7R3 72703685 IC50 = 250 nM T84621 CAU4Z0 72703889 IC50 = 1010 nM T84621 C56KEC 72703890 IC50 = 1480 nM T84621 C4AEX3 73347616 IC50 = 38 nM T84621 CFD46C 73347617 IC50 = 5 nM T84621 C26LJW 73347618 IC50 = 1015 nM T84621 CIHF35 73350707 IC50 = 51 nM T84621 CT26EZ 73355186 IC50 > 5000 nM T84621 C0NXU4 73355187 IC50 = 87 nM T84621 CML29U 73355188 IC50 = 427 nM T84621 CC5TO4 73356735 IC50 = 125 nM T84621 CWZ3A1 73356736 IC50 = 1.3 nM T84621 C9CY3K 73442767 IC50 = 34 nM T84621 CU6IQ9 73603293 IC50 = 4737 nM T84621 C6MQ8L 73603294 IC50 > 5000 nM T84621 CR81XZ 73603295 IC50 = 1423 nM T84621 CJS6Y2 73603296 IC50 > 5000 nM T84621 C1GR7W 73603297 IC50 > 5000 nM T84621 CM4L6N 73603298 IC50 = 1523 nM T84621 CAIB62 73603299 IC50 > 5000 nM T84621 C7G6KZ 73603343 IC50 = 52 nM T84621 CDX9R1 73603344 IC50 = 516 nM T84621 C7KV2S 73603345 IC50 = 6093 nM T84621 CM10ZX 73603346 IC50 = 3723 nM T84621 CJSY07 73603348 IC50 = 1379 nM T84621 CS03UP 73603349 IC50 = 6812 nM T84621 C56LYP 73603350 IC50 = 6642 nM T84621 C9RKH0 73603387 IC50 = 803 nM T84621 CG86BD 73603388 IC50 = 3125 nM T84621 C2R3ZB 73603389 IC50 = 3756 nM T84621 C5ARE7 73603390 IC50 = 160 nM T84621 CTMF86 73603391 IC50 = 366 nM T84621 C5RG4C 75593332 IC50 = 10.74 nM T84621 CMN51L 76286753 IC50 > 8300 nM T84621 C06HYT 76286902 IC50 = 1299 nM T84621 CPU3T6 76317295 IC50 = 7.2 nM T84621 CZ2U9K 76321000 IC50 = 1.5 nM T84621 C4UO5H 76331904 IC50 < 0.1 nM T84621 CP10SN 76335488 IC50 = 0.3 nM T84621 C1YJW0 77846787 IC50 = 32 nM T84621 CV73PD 77846790 IC50 = 82 nM T84621 C0DIH7 77846872 IC50 = 17 nM T84621 COI25M 77846873 IC50 = 67 nM T84621 CJI8R0 77846875 IC50 = 29 nM T84621 CZK4J1 77846962 IC50 = 70 nM T84621 CEK89G 77846963 IC50 = 110 nM T84621 C5BA8Z 77846964 IC50 = 187 nM T84621 C4D6XJ 77847803 IC50 = 63 nM T84621 CF7O4Q 77847804 IC50 = 40 nM T84621 C2ASY0 86730379 IC50 = 880 nM T84621 CA4QV9 86730380 IC50 = 33 nM T84621 C24ZMT 86730381 IC50 = 37 nM T84621 C9W6RO 86730382 IC50 = 600 nM T84621 C3UMP9 89471867 IC50 = 640 nM T84621 CW8TF6 89471869 IC50 = 300 nM T84621 CL30TR 89471870 IC50 = 760 nM T84621 CJ0H5V 89471872 IC50 = 1100 nM T84621 C3BUS8 89471889 IC50 = 930 nM T84621 CI7HY8 89471890 IC50 = 800 nM T84621 CF2AY7 89471891 IC50 > 8700 nM T84621 CQF07X 89471892 IC50 = 830 nM T84621 C62KFZ 89961587 IC50 > 10000 nM T84621 C8XS2I 89961629 IC50 = 317 nM T84621 C75PMO 89961672 IC50 > 8333 nM T84621 CX0M7B 89961716 IC50 = 1357 nM T84621 C3JN5I 89961721 IC50 > 10000 nM T84621 CSJT14 89961765 IC50 = 1473 nM T84621 CR5D6Y 89961785 IC50 > 10000 nM T84621 C7TI3V 89961787 IC50 > 8333 nM T84621 C2QP7I 89961848 IC50 > 10000 nM T84621 C81FEN 89961879 IC50 > 10000 nM T84621 CI6P0R 89961978 IC50 > 8333 nM T84621 C89TEU 89968659 IC50 = 5705 nM T84621 C7BC5N 89968688 IC50 > 10000 nM T84621 C3XIF5 90252771 IC50 = 1.1 nM T84621 CGZ2S1 90252806 IC50 = 470 nM T84621 C4F9VB 90252809 IC50 = 1400 nM T84621 CE2TM0 90252810 IC50 > 8300 nM T84621 CGVL78 90252811 IC50 > 8300 nM T84621 C0S3HV 90252812 IC50 = 916 nM T84621 C4M8TO 90252814 IC50 = 1200 nM T84621 CM0T2X 90252815 IC50 > 8300 nM T84621 CY5IC7 90252834 IC50 = 98 nM T84621 CF05JI 90252835 IC50 = 1000 nM T84621 C72ICB 90252839 IC50 > 8300 nM T84621 C84NVA 90252850 IC50 = 338 nM T84621 CBY46O 90252851 IC50 = 856 nM T84621 CNVA50 90252852 IC50 = 386 nM T84621 C0Z2TI 90252864 IC50 = 47 nM T84621 CV30CD 90252953 IC50 = 535 nM T84621 C3MV7S 90252954 IC50 = 1690 nM T84621 CD5ST8 90252956 IC50 > 8300 nM T84621 C3JH4P 90252957 IC50 > 8300 nM T84621 CCU4F7 90252958 IC50 = 1987 nM T84621 C89BFG 90333640 IC50 = 58 nM T84621 C82YUB 90644545 IC50 = 302 nM T84621 CVFA18 90644546 IC50 = 736 nM T84621 CR50EN 90644547 IC50 = 61 nM T84621 C46ZNM 90644548 IC50 = 435 nM T84621 CS6N1P 90644549 IC50 = 4100 nM T84621 CB5HI4 90644550 IC50 = 2300 nM T84621 CHD21I 90666137 IC50 = 21.2 nM T84621 CLB2E7 91827654 IC50 = 4402 nM T84621 C5GV1L 101882447 IC50 = 5 nM T84621 CMH51N 118496543 IC50 = 779 nM T84621 C3ZPQ1 118496545 IC50 = 149 nM T84621 CJ9Z0S 118496546 IC50 = 22 nM T84621 C7UN3R 118496547 IC50 = 197 nM T84621 CJ54UQ 118618017 IC50 = 872 nM T84621 CLS25A 118714825 IC50 = 111 nM T84621 CT0FH7 118714826 IC50 = 327 nM T84621 CD8T1P 118714827 IC50 = 1674 nM T84621 C85BVO 118714828 IC50 = 690 nM T84621 CYFP62 118714829 IC50 = 499 nM T84621 CE3ZF1 118714830 IC50 = 2003 nM T84621 C5HKE1 118714831 IC50 = 1750 nM T84621 C7BD3X 118714832 IC50 = 587 nM T84621 C9BM7X 118714833 IC50 = 188 nM T84621 CML4K7 118714834 IC50 = 68 nM T84621 CE5L8U 118714835 IC50 = 2001 nM T84621 CD8YA9 118714836 IC50 > 5000 nM T84621 CRNL64 118714837 IC50 = 28 nM T84621 C4F6AY 118714838 IC50 = 65 nM T84621 CZ9L5S 118714839 IC50 = 334 nM T84621 CU3XP2 118714840 IC50 = 26 nM T84621 C0BRP1 118714841 IC50 = 278 nM T84621 C6M5VU 118714842 IC50 = 382 nM T84621 CQ5KI0 118714843 IC50 = 929 nM T84621 C32MDK 118714844 IC50 = 71 nM T84621 C15PAW 118714845 IC50 = 49 nM T84621 CPH51S 118714846 IC50 = 62 nM T84621 C1L4YZ 118714847 IC50 = 137 nM T84621 CLM64U 118714848 IC50 = 309 nM T84621 C5UD3K 118714849 IC50 = 1224 nM T84621 CNW8E3 118714850 IC50 = 65 nM T84621 CMXG03 118714851 IC50 = 114 nM T84621 CTWO23 118714852 IC50 = 60 nM T84621 CAW36P 118714853 IC50 = 663 nM T84621 C4Y2UF 118714854 IC50 = 1167 nM T84621 CJK08Q 118714855 IC50 = 6 nM T84621 CP4O0C 118720463 IC50 = 6712 nM T84621 CV4IC9 118720464 IC50 = 4196 nM T84621 CKG28R 118720465 IC50 = 7315 nM T84621 CGXD81 118720466 IC50 = 1096 nM T84621 CF1W7I 118720467 IC50 = 8947 nM T84621 COZU39 118720468 IC50 = 4797 nM T84621 CWG6L8 118720469 IC50 = 4487 nM T84621 C2HV3Y 118720470 IC50 = 5549 nM T84621 CX56BZ 118720471 IC50 = 6548 nM T84621 CO8H3J 118720472 IC50 = 7427 nM T84621 C7WEQ3 118720473 IC50 = 5812 nM T84621 CG8PB5 118720474 IC50 = 4710 nM T84621 CN2U6B 118720475 IC50 = 6189 nM T84621 CU7FW1 118720476 IC50 = 6674 nM T84621 CCJ17Z 118720477 IC50 = 5076 nM T84621 CB4DS9 118720479 IC50 = 8550 nM T84621 CC9V6K 118720480 IC50 = 8333 nM T84621 CP7X1B 118720481 IC50 = 9346 nM T84621 CPT58L 118720482 IC50 = 4717 nM T84621 C3E7TA 118720483 IC50 = 6534 nM T84621 CS01NU 118720484 IC50 = 6164 nM T84621 CAW5K3 118723935 IC50 = 48 nM T84621 CK8UL1 118723936 IC50 = 111 nM T84621 CIW7O0 118723937 IC50 = 63 nM T84621 C42CEZ 118723938 IC50 = 48 nM T84621 CJQ63E 118723939 IC50 = 258 nM T84621 CCXN71 118723940 IC50 = 57 nM T84621 CS78BD 118723941 IC50 = 50 nM T84621 C9W3QX 118723942 IC50 > 500 nM T84621 COJ2K8 118723943 IC50 = 15 nM T84621 CZ23UL 118723944 IC50 = 24 nM T84621 CIWU64 118723945 IC50 = 30 nM T84621 CZI6A0 118723946 IC50 = 109 nM T84621 COB46M 118723947 IC50 = 518 nM T84621 CYM08W 118726850 IC50 = 120 nM T84621 CR32JU 118726851 IC50 = 4.5 nM T84621 C2OAI6 118726852 IC50 = 7483 nM T84621 CDHI10 118733086 IC50 > 10000 nM T84621 C18PWB 118733087 IC50 > 10000 nM T84621 C8WJ2Y 118733088 IC50 > 10000 nM T84621 C31ZXP 118733089 IC50 > 10000 nM T84621 CHR84E 118733090 IC50 > 10000 nM T84621 CAQ72M 118733091 IC50 > 10000 nM T84621 CIV1Z5 118733092 IC50 > 10000 nM T84621 CU3Y9W 118733093 IC50 > 10000 nM T84621 CF49NU 118733094 IC50 > 10000 nM T84621 CK73VU 118733095 IC50 > 10000 nM T84621 CR1WU5 118733096 IC50 > 10000 nM T84621 C1V7WI 118735163 IC50 = 279 nM T84621 C6YG9R 118735164 IC50 = 1207 nM T84621 C5C4FZ 118735165 IC50 = 540 nM T84621 C1ZLM6 118735166 IC50 = 23 nM T84621 CQXM57 118735167 IC50 = 13 nM T84621 C0RYM4 118735168 IC50 = 6 nM T84621 C0DCB9 118735169 IC50 = 50 nM T84621 CG4QF3 118735170 IC50 = 2 nM T84621 CD3IY5 118735171 IC50 = 8 nM T84621 C0JZ2Y 118735172 IC50 = 508 nM T84621 C2WS7A 118735173 IC50 = 1201 nM T84621 CYEA24 118735174 IC50 = 51 nM T84621 CZ9X4J 118735175 IC50 = 60 nM T84621 CG14RD 118735176 IC50 = 183 nM T84621 CQ3KR4 118735177 IC50 = 46 nM T84621 C1Z9FX 118735178 IC50 = 812 nM T84621 C2VJU4 118735179 IC50 = 26 nM T84621 CXWH51 118735180 IC50 = 38 nM T84621 C3YUS9 118735181 IC50 = 12 nM T84621 CEH97S 118735182 IC50 = 594 nM T84621 C03HKR 118735183 IC50 = 1150 nM T84621 CC38HG 118735184 IC50 = 1665 nM T84621 C8QIC4 118735185 IC50 = 2665 nM T84621 CZET62 118735186 IC50 = 182 nM T84621 CZ8U2C 118735187 IC50 = 6 nM T84621 CUAE09 121004872 IC50 > 8333 nM T84621 C1OT4E 121458684 IC50 = 1552 nM T84621 C9ETN3 121458685 IC50 = 795 nM T84621 C4V2HU 121458987 IC50 = 225 nM T84621 CPGD72 121458994 IC50 = 117 nM T84621 CXW13O 122179553 IC50 > 10000 nM T84621 C3E0VM 122179554 IC50 > 10000 nM T84621 CJVX13 122179555 IC50 > 8333 nM T84621 CWN9K7 122179556 IC50 > 10000 nM T84621 CV2PQ1 122191831 IC50 > 8333 nM T84621 C2AHB5 122191832 IC50 > 8333 nM T84621 CFZH01 122191833 IC50 > 8333 nM T84621 C1XKA8 122191834 IC50 > 8333 nM T84621 CG4S8F 122191835 IC50 = 887 nM T84621 C37NLK 122191836 IC50 > 8333 nM T84621 CVT7A2 127027254 IC50 = 86.9 nM T84621 C5QNG6 127027265 IC50 > 10000 nM T84621 CIZO64 127027266 IC50 > 10000 nM T84621 C9RXH3 127027267 IC50 > 10000 nM T84621 CEM84R 127027569 IC50 = 1600.8 nM T84621 CT83ZE 127027570 IC50 = 326.9 nM T84621 CHZ54G 127027571 IC50 = 29.5 nM T84621 C2ZFR8 127027572 IC50 = 108.9 nM T84621 CV1BD6 127027573 IC50 = 9.7 nM T84621 C0E6DW 127027574 IC50 > 10000 nM T84621 C2MFJ8 127027575 IC50 > 10000 nM T84621 CM8T9G 127028498 IC50 = 612.3 nM T84621 CQO36B 127028499 IC50 = 58.1 nM T84621 C1M7GD 127028500 IC50 = 222.5 nM T84621 CN42BR 127028817 IC50 = 82.7 nM T84621 C3IMJ8 127028818 IC50 = 179.6 nM T84621 CPEM69 127028819 IC50 = 372.1 nM T84621 C70XOB 127030295 IC50 = 3598.4 nM T84621 CZ7L4J 127031191 IC50 > 10000 nM T84621 C49IME 127031799 IC50 = 88.2 nM T84621 CHS8L7 131982520 IC50 = 1900 nM T84621 C95PYQ 131982530 IC50 = 350 nM T84621 C5IWD9 131982539 IC50 = 2400 nM T84621 CSIP72 131982576 IC50 < 100 nM T84621 CS8C7T 131982729 IC50 = 1100 nM T84621 CHDP80 131982862 IC50 = 410 nM T84621 C1BNU6 131982871 IC50 > 10000 nM T84621 C6CB0I 132585204 IC50 = 2 nM T84621 C7SM9W 134129925 IC50 = 387 nM T84621 CB3EL1 134134056 IC50 = 1595 nM T84621 CB79AO 134134186 IC50 = 1308 nM T84621 CPZX32 134135994 IC50 = 10000 nM T84621 CS2P0E 134136577 IC50 = 2192 nM T84621 CH3V9Q 134139925 IC50 = 460 nM T84621 CFUE13 134141128 IC50 = 1573 nM T84621 COUK40 134141967 IC50 = 1996 nM T84621 CX3Y9D 134142597 IC50 = 1674 nM T84621 CQF59S 134143092 IC50 = 787 nM T84621 C1HG8V 134144349 IC50 = 1739 nM T84621 CFC8O6 134145376 IC50 = 220 nM T84621 C31WNO 134145695 IC50 > 8000 nM T84621 C7JEU2 134148873 IC50 = 250 nM T84621 C2JOB5 134152002 IC50 = 1544 nM T84621 CTXL17 134153274 IC50 = 1000 nM T84621 C3OLF2 134153424 IC50 > 8000 nM T84621 C12LPH 134153935 IC50 = 355 nM T84621 C8ROI0 134153997 IC50 = 630 nM T84621 CDV8M5 134155385 IC50 = 4600 nM T84621 C74ONC 134156861 IC50 = 4460 nM T84621 CKL9N7 135185757 IC50 = 4629 nM T84621 C8HTS7 135185761 IC50 > 10000 nM T84621 C1D4CS 135185764 IC50 = 5380 nM T84621 CMQC50 135185766 IC50 = 378 nM T84621 CIS5H8 135185771 IC50 = 4157 nM T84621 CF0EC1 135185786 IC50 = 4325 nM T84621 C8GB5V 135185787 IC50 = 2035 nM T84621 CH30EN 135185789 IC50 = 3330 nM T84621 CMR5C9 135185792 IC50 = 3926 nM T84621 CX97YM 135185793 IC50 = 1907 nM T84621 CS5FX2 135185796 IC50 = 2267 nM T84621 CV9RM5 135185801 IC50 = 4987 nM T84621 C8MF2Z 135185815 IC50 = 390 nM T84621 CX57GP 135185833 IC50 = 4809 nM T84621 CSZA19 135185836 IC50 = 5723 nM T84621 C6G1CH 135185858 IC50 = 4771 nM T84621 C9LU0C 135185886 IC50 = 4171 nM T84621 CZ1JS3 135186252 IC50 > 10000 nM T84621 CWU63C 136008115 IC50 = 17 nM T84621 CAV9U3 136219390 IC50 = 230 nM T84621 CC7LY3 136239517 IC50 = 960 nM T84621 C2V0IM 136244612 IC50 = 75 nM T84621 CYIF59 136245971 IC50 > 5000 nM T84621 CM97FH 137631528 IC50 = 48 nM T84621 C9LY0O 137631806 IC50 = 1 nM T84621 CH05YR 137633095 IC50 = 20 nM T84621 COG72W 137633343 IC50 = 93 nM T84621 C3QE1V 137633417 IC50 = 3 nM T84621 CVM54L 137634483 IC50 = 4 nM T84621 CV2S5Q 137637282 IC50 = 110 nM T84621 CUIX95 137637496 IC50 = 210 nM T84621 C14LXC 137638585 IC50 = 13 nM T84621 C1D0WG 137638612 IC50 = 9 nM T84621 CF1D5C 137639549 IC50 = 11 nM T84621 C8V7CD 137639692 IC50 = 6 nM T84621 C1SH2M 137639834 IC50 = 1.8 nM T84621 CZA2S8 137639890 IC50 = 14 nM T84621 C0N4PJ 137640302 IC50 = 124 nM T84621 COEV02 137642385 IC50 = 16 nM T84621 CH35RE 137642529 IC50 = 0.6 nM T84621 CP1EJ0 137642735 IC50 = 22 nM T84621 C29FMO 137642787 IC50 = 137 nM T84621 COGQ01 137644314 IC50 = 16 nM T84621 CA73KP 137644560 IC50 = 150 nM T84621 C4UP3J 137647900 IC50 = 2 nM T84621 CI31EQ 137649226 IC50 = 516 nM T84621 CS5BW7 137650545 IC50 = 4 nM T84621 CF71RE 137650772 IC50 = 104 nM T84621 CQ54YG 137651298 IC50 = 5 nM T84621 C4CL2W 137651728 IC50 = 42 nM T84621 CK7QJ4 137651744 IC50 = 2 nM T84621 CI5D2P 137652926 IC50 = 5 nM T84621 CIH34U 137653629 IC50 = 520 nM T84621 CV9I5G 137653991 IC50 = 13 nM T84621 C28VRO 137654883 IC50 = 19 nM T84621 CEV94S 137655303 IC50 = 148 nM T84621 CY5IK7 137655531 IC50 = 2 nM T84621 CUL37V 137655879 IC50 = 1 nM T84621 CN2CQ1 137656473 IC50 = 62 nM T84621 C53NVI 137657989 IC50 = 3 nM T84621 CNI0C1 137658011 IC50 = 42 nM T84621 C32WHO 137658276 IC50 = 181 nM T84621 C0G2UI 137658690 IC50 = 58 nM T84621 CLNU74 137659288 IC50 = 57 nM T84621 CA5LI1 137659926 IC50 = 14 nM T84621 C7YI9N 137660712 IC50 = 10 nM T84621 CFU1Z3 145960404 IC50 = 130 nM T84621 C1IU5W 145960520 IC50 = 1200 nM T84621 CQFH90 145960862 IC50 = 590 nM T84621 CNIB73 145960902 IC50 = 480 nM T84621 C0KNY4 145961099 IC50 < 100 nM T84621 CGI39P 145961215 IC50 = 2100 nM T84621 CW84OQ 145961259 IC50 > 10000 nM T84621 C92JOV 145961758 IC50 > 10000 nM T84621 CR6JH8 145961916 IC50 = 2200 nM T84621 CS4EO5 145962296 IC50 = 180 nM T84621 C1O0NQ 145962517 IC50 = 5700 nM T84621 C6VO0A 145962577 IC50 < 100 nM T84621 CY20CQ 145962664 IC50 > 10000 nM T84621 C6F7UE 145962949 IC50 = 58 nM T84621 C5O4RQ 145963242 IC50 > 10000 nM T84621 CGA01F 145963470 IC50 = 470 nM T84621 CH0TM7 145963574 IC50 > 10000 nM T84621 C0TZR1 145964456 IC50 = 19.2 nM T84621 CRJM82 145965429 IC50 = 6.6 nM T84621 CN7B1I 145968025 IC50 = 12.3 nM T84621 C82JTH 145971322 IC50 = 11.4 nM T84621 C5R6SH 145973507 IC50 = 5.8 nM T84621 C41LQE 145976039 IC50 = 4.7 nM T84621 C01TYI 145976345 IC50 = 15.4 nM T84621 CG23BW 145977901 IC50 = 6.5 nM T84621 C65ZFY 145978611 IC50 = 4.1 nM T84621 CI48QV 145979205 IC50 = 77 nM T84621 C9IQK7 145980859 IC50 = 17 nM T84621 CCKL25 145981178 IC50 = 120 nM T84621 CY4G3E 145981780 IC50 = 0.8 nM T84621 CYI3V5 145988023 IC50 = 29 nM T84621 CH6DJ3 155527950 IC50 = 4523 nM T84621 C80XNT 155530085 IC50 = 1668 nM T84621 C5XB1F 155530577 IC50 > 10000 nM T84621 C6DXN8 155559405 IC50 > 10000 nM T84621 C4UQS2 155564575 IC50 > 10000 nM T84621 CXM62E 155566406 IC50 = 9072 nM T84621 D00BVP 11847320 IC50 = 7 nM T84621 D00DSE 49864196 IC50 = 928 nM T84621 D00DUJ 11687499 IC50 = 7553 nM T84621 D00PXF 44206698 IC50 = 32.36 nM T84621 D01JZO 2779191 IC50 = 1000 nM T84621 D01REI 46901610 IC50 = 1400 nM T84621 D01SUE 6539759 IC50 = 888 nM T84621 D01SZX 46867545 IC50 = 99.1 nM T84621 D02ALK 11514074 IC50 = 2671 nM T84621 D02BXS 46901445 IC50 = 902 nM T84621 D02CSU 6539786 IC50 = 931 nM T84621 D02GFK 25034431 IC50 = 1521 nM T84621 D02JUJ 25034344 IC50 = 8925 nM T84621 D02LWB 6540046 IC50 = 2391 nM T84621 D02NAG 6539765 IC50 = 1472 nM T84621 D02PSL 45103913 IC50 = 6.166 nM T84621 D02UZI 6540056 IC50 = 288 nM T84621 D02XHH 6540043 IC50 = 23.5 nM T84621 D02ZQM 25180104 IC50 = 4921 nM T84621 D03CWL 14535954 IC50 = 323.59 nM T84621 D03EXD 49864181 IC50 = 251 nM T84621 D03KLN 11413434 IC50 = 81 nM T84621 D03MKT 6539788 IC50 = 1098 nM T84621 D03TRM 6540032 IC50 = 25.9 nM T84621 D03VRC 2989557 IC50 = 211 nM T84621 D03YHZ 25147692 IC50 = 33 nM T84621 D04CFP 46901927 IC50 = 469 nM T84621 D04CLL 6539775 IC50 = 763 nM T84621 D04ELJ 6539766 IC50 = 270 nM T84621 D04IBH 11616637 IC50 = 4481 nM T84621 D04ISG 11680597 IC50 = 2724 nM T84621 D04PKP 23644953 IC50 = 2896 nM T84621 D04QPK 6539783 IC50 = 774 nM T84621 D04WJN 10588478 IC50 = 70.8 nM T84621 D05FFY 14231155 IC50 = 141 nM T84621 D05IXU 25130517 IC50 = 953 nM T84621 D05MQE 6539785 IC50 = 657 nM T84621 D05QPR 12229388 IC50 = 489.78 nM T84621 D06CWR 24754344 IC50 = 67 nM T84621 D06HFV 6539805 IC50 = 27 nM T84621 D06JYY 25130848 IC50 = 2804 nM T84621 D06NFC 45103808 IC50 = 16 nM T84621 D06RSD 45103911 IC50 = 307 nM T84621 D07CTI 10853186 IC50 = 22.3 nM T84621 D07DQJ 45103810 IC50 = 7 nM T84621 D07EJK 10632289 IC50 = 478 nM T84621 D07IQG 10473365 IC50 = 6.7 nM T84621 D07JCO 12354256 IC50 = 6338 nM T84621 D07JMO 10220337 IC50 = 143 nM T84621 D07NAH 21772021 IC50 = 207 nM T84621 D07PYC 6539760 IC50 = 87 nM T84621 D07SOM 11847316 IC50 = 12 nM T84621 D07VGT 46901929 IC50 = 627 nM T84621 D07WLT 25180108 IC50 = 3964 nM T84621 D08AZK 6539767 IC50 = 1937 nM T84621 D08EZA 11847317 IC50 = 187 nM T84621 D08FAB 11845485 IC50 = 5826 nM T84621 D08HHA 19902087 IC50 = 204.17 nM T84621 D08HPU 6540052 IC50 = 503 nM T84621 D08IDC 24827305 IC50 = 238 nM T84621 D08ORG 10198247 IC50 = 281.84 nM T84621 D08PNF 6539770 IC50 = 790 nM T84621 D08WHC 10397593 IC50 = 206 nM T84621 D08YGW 10444038 IC50 = 4.786 nM T84621 D08ZTZ 11529133 IC50 = 2517 nM T84621 D09CPC 13728862 IC50 = 6746 nM T84621 D09HEA 1236449 IC50 = 368 nM T84621 D09HOE 6539789 IC50 = 34 nM T84621 D09QDY 6540033 IC50 = 6.1 nM T84621 D09VPA 6539794 IC50 = 2640 nM T84621 D09VQZ 46901616 IC50 = 4742 nM T84621 D09YXV 6539769 IC50 = 1448 nM T84621 D09ZHX 11847318 IC50 = 27 nM T84621 D0AK9S 22466877 IC50 = 18 nM T84621 D0AW7Q 46867544 IC50 = 463 nM T84621 D0B2UM 25034430 IC50 = 114 nM T84621 D0C6US 6540055 IC50 = 2529 nM T84621 D0C7YL 6481821 IC50 = 390 nM T84621 D0D7YL 11586681 IC50 = 2452 nM T84621 D0D8KN 45103805 IC50 = 181 nM T84621 D0D8YE 6540048 IC50 = 5684 nM T84621 D0D9FR 6539795 IC50 = 484 nM T84621 D0E0ZS 46901613 IC50 = 307 nM T84621 D0E8DX 25180300 IC50 = 580 nM T84621 D0E9WX 6540042 IC50 = 26.2 nM T84621 D0F5AC 46867542 IC50 = 15.1 nM T84621 D0F5YU 6539793 IC50 = 301 nM T84621 D0G6QL 23644748 IC50 = 1317 nM T84621 D0G9WP 18407230 IC50 = 819 nM T84621 D0HL9S 1265319 IC50 = 234.42 nM T84621 D0I1YH 46901446 IC50 = 342 nM T84621 D0I2UH 44187006 IC50 = 5.754 nM T84621 D0I5NW 6540047 IC50 = 1729 nM T84621 D0I9PA 25180306 IC50 = 13378 nM T84621 D0JE1I 9815923 IC50 = 9.5 nM T84621 D0K2DR 12050204 IC50 = 5952 nM T84621 D0K5KG 6540050 IC50 = 1268 nM T84621 D0L2QD 45103910 IC50 = 72.44 nM T84621 D0L4NG 6540054 IC50 = 1615 nM T84621 D0L8KL 11275595 IC50 = 805 nM T84621 D0LJ9D 46901783 IC50 = 415 nM T84621 D0M7FS 6539764 IC50 = 125 nM T84621 D0M9VK 11514098 IC50 = 849 nM T84621 D0MA9G 6540051 IC50 = 2117 nM T84621 D0N1GH 11601068 IC50 = 691 nM T84621 D0N1PQ 11506923 IC50 = 1577 nM T84621 D0N4VI 3021558 IC50 = 639 nM T84621 D0N5GZ 12229395 IC50 = 258 nM T84621 D0N8QD 15594569 IC50 = 691.83 nM T84621 D0N9PY 6539773 IC50 = 2368 nM T84621 D0NV7W 45103912 IC50 = 19.95 nM T84621 D0NX0M 6540049 IC50 = 578 nM T84621 D0O7TC 25180103 IC50 = 525 nM T84621 D0P1UO 45103914 IC50 = 26.92 nM T84621 D0PH1G 13688208 IC50 = 47.86 nM T84621 D0Q0BK 46901611 IC50 = 850 nM T84621 D0Q3CX 25034343 IC50 = 52 nM T84621 D0Q3JZ 6539774 IC50 = 2697 nM T84621 D0Q5ZZ 25129117 IC50 = 640 nM T84621 D0Q6BJ 25034426 IC50 = 151 nM T84621 D0Q8KM 44206482 IC50 = 28 nM T84621 D0R0TE 11557864 IC50 = 5419 nM T84621 D0RJ6S 11558270 IC50 = 2939 nM T84621 D0S4KP 25034427 IC50 = 843 nM T84621 D0S4WQ 12229386 IC50 = 151.36 nM T84621 D0S8FV 44586852 IC50 = 1047 nM T84621 D0T8JU 45103811 IC50 = 10.96 nM T84621 D0U7RR 6539768 IC50 = 320 nM T84621 D0V3YH 6539784 IC50 = 304 nM T84621 D0V6QN 45103915 IC50 = 128.82 nM T84621 D0V8CR 6539763 IC50 = 311 nM T84621 D0VL3R 25180303 IC50 = 1977 nM T84621 D0W8IZ 45103809 IC50 = 25.12 nM T84621 D0WN9P 46901444 IC50 = 287 nM T84621 D0X0IH 77918 IC50 = 135 nM T84621 D0X1QS 6540053 IC50 = 1291 nM T84621 D0Y3AV 25034346 IC50 = 373 nM T84621 D0Y5KX 46901443 IC50 = 522 nM T84621 D0YD9J 6539792 IC50 = 1515 nM T84621 D0YS2F 6539776 IC50 = 955 nM T84621 D0Z3GX 46901784 IC50 = 422 nM T35173 D03MXK 25022340 Ki = 5.1 nM T35173 D07CLV 46940575 IC50 = 12.9 nM T35173 D09MIN 24737642 IC50 = 11 nM T35173 D08XOV 50913339 IC50 = 1.3 nM T35173 D0YN1X 71661892 Ki = 5.4 nM T35173 CO1ZE4 9927170 IC50 = 690 nM T35173 CY3RV2 17756618 Ki = 2 nM T35173 CBM94F 23646361 Ki = 328 nM T35173 C8XJG1 24754961 Ki > 10000 nM T35173 C3EN8I 24857831 IC50 = 1860 nM T35173 C7XTN2 25138055 Ki = 5.9 nM T35173 CJ2VZ4 25138056 Ki = 4.2 nM T35173 C29PBM 25138057 Ki = 370 nM T35173 CLO6Y8 25138058 Ki = 20 nM T35173 CPN8E5 25138069 Ki = 1 nM T35173 CWH17B 25138070 Ki = 132 nM T35173 C0BJQ6 25173661 Ki = 20800 nM T35173 CW4U0R 25180313 Ki = 3 nM T35173 CAL8M3 25209021 Ki = 0.25 nM T35173 CD29TU 25209022 Ki = 2.09 nM T35173 C2KPJ0 44576646 IC50 = 1890 nM T35173 C96OTK 46830178 Ki = 24 nM T35173 CECL56 46830179 Ki = 393 nM T35173 C8RDC3 46888403 Ki = 292 nM T35173 CP40QG 46929436 Ki = 4.2 nM T35173 CQ0A5I 46929438 Ki = 47 nM T35173 C5FK8W 46929440 IC50 = 5.3 nM T35173 C1TIK8 46930628 Ki = 22.5 nM T35173 CVC3T5 46930723 Ki = 24.8 nM T35173 CNQO70 52951104 Ki = 1.7 nM T35173 C30GIF 53237922 Ki = 6 nM T35173 CW7AF2 53238154 Ki = 2 nM T35173 C5JPH2 53238155 Ki = 1.2 nM T35173 CW71DY 53238387 Ki = 2 nM T35173 C16JNG 53238388 Ki = 3 nM T35173 C3IPJ4 53238615 Ki = 2 nM T35173 CH0L8C 53238616 Ki = 2 nM T35173 CF83PC 53238842 Ki = 2.5 nM T35173 C2HB0C 53238843 Ki = 3 nM T35173 C7SR2W 53239063 Ki = 2.5 nM T35173 CM46PV 53239064 Ki = 4 nM T35173 CNFD80 53239285 Ki = 7 nM T35173 CCL6I5 53239286 Ki = 11 nM T35173 C61NHL 56945169 Ki = 3.3 nM T35173 C2WXP5 56945170 Ki = 6.4 nM T35173 C7YW1J 56945269 Ki = 6.9 nM T35173 CR7TD9 56945270 Ki = 14 nM T35173 CAD3P5 56945392 Ki = 4 nM T35173 CDYL09 56945393 Ki = 11 nM T35173 C7X1ZF 56946798 Ki = 1.7 nM T35173 C05JAE 56946799 Ki = 1.3 nM T35173 CE6SU4 57689264 Ki = 2 nM T35173 C62ZCQ 57689338 Ki = 25.3 nM T35173 C3KDR0 58609608 IC50 = 209 nM T35173 CTYP01 66972671 IC50 = 2.6 nM T35173 CZI6S5 66972777 IC50 = 4 nM T35173 CK0FP7 66972990 IC50 = 2.7 nM T35173 CQ9Y8K 66972994 IC50 = 3.2 nM T35173 CTKN28 66973039 IC50 = 2.5 nM T35173 CR9CO4 66973072 IC50 = 3.4 nM T35173 CKQ68O 66973165 IC50 = 4.9 nM T35173 CAD24O 66973224 IC50 = 7.6 nM T35173 C0R9TP 66973397 IC50 = 14 nM T35173 CQ1O6Z 66973400 IC50 = 2.1 nM T35173 C1NV7Q 71528757 EC50 = 36 nM T35173 C5RD4E 71570901 IC50 = 214 nM T35173 C9IT5Y 71570902 IC50 = 235 nM T35173 CY83OB 71571046 EC50 = 20 nM T35173 CAR8J2 71578011 IC50 = 1320 nM T35173 CVPJ20 71581702 IC50 = 47 nM T35173 CP9G3R 71581703 IC50 = 11 nM T35173 C3F4OT 71581838 IC50 = 40 nM T35173 CLIU93 71582189 IC50 = 16 nM T35173 C1VME6 71582339 IC50 = 10 nM T35173 CZ8DF4 71661893 Ki = 12.6 nM T35173 CB0O2T 71662077 Ki = 7.7 nM T35173 COCI81 71662078 Ki = 9.9 nM T35173 CNU16X 71662256 Ki = 2.1 nM T35173 CJRL34 71662257 Ki = 10 nM T35173 C2UM5A 71662420 Ki = 11 nM T35173 CVZK59 71662421 Ki = 7.4 nM T35173 CW4G0O 71662584 Ki = 13.3 nM T35173 C8AY6G 71662585 Ki = 7.9 nM T35173 C2UVF7 76335647 IC50 = 21 nM T35173 CZQO17 86650974 IC50 = 1.7 nM T35173 C9PHL5 89569624 IC50 = 24 nM T35173 CO0IY8 89570499 IC50 = 232 nM T35173 CD57CO 89570570 IC50 = 1490 nM T35173 C2ARB5 89570664 IC50 = 900 nM T35173 CIH2F9 90657109 IC50 = 366 nM T35173 CIH5V8 90664859 IC50 = 1300 nM T35173 C7APL4 118732792 IC50 = 1360 nM T35173 CDZ6M0 118732793 IC50 = 2880 nM T35173 C64NWU 118732794 IC50 = 180 nM T35173 CI69WD 118732795 IC50 = 17 nM T35173 C14FGL 122187534 IC50 = 3 nM T35173 C6NFD0 134419123 IC50 = 330 nM T35173 C87BOG 138377561 IC50 = 5.7 nM T35173 C0B8GK 138377594 IC50 = 140 nM T35173 CA43ML 142585287 IC50 > 1000 nM T35173 CGF6R2 142585309 IC50 > 1000 nM T35173 C0HC8R 142585337 IC50 > 9000 nM T35173 C0RHF1 142585361 IC50 > 10000 nM T35173 C5AI8Z 142585365 IC50 > 10000 nM T35173 CM7IG2 142585375 IC50 > 1500 nM T35173 CG46IU 145954838 IC50 > 1000 nM T35173 CKEJ30 145979040 IC50 = 353.3 nM T35173 C7XM4Q 145979112 IC50 = 53.5 nM T35173 CLRM52 145979809 IC50 = 304 nM T35173 CL4F9B 145981512 IC50 = 1103 nM T35173 C1K6AY 145982930 IC50 > 1000 nM T35173 C3L1ZW 145985393 IC50 = 56.6 nM T35173 CY8JR0 145986444 IC50 = 364.3 nM T35173 C1HWA3 145988725 IC50 = 212.1 nM T35173 CX7AV2 145991404 IC50 = 30.6 nM T35173 C79EXP 145992527 IC50 = 15 nM T35173 CK8JB2 155512591 IC50 = 40 nM T35173 CEH0W4 155523271 IC50 = 353 nM T35173 C23UZA 155554597 IC50 = 12.5 nM T35173 CR3UQ4 155561157 IC50 = 9 nM T35173 D03KZH 25172871 Ki = 6.3 nM T35173 D0BW7P 44589292 Ki = 4.8 nM T35173 D0Q7TL 24754886 Ki = 1.84 nM T35173 D0VK7M 49847690 IC50 = 21 nM T91442 D05RQB 457964 IC50 = 600 nM T91442 CZP5J2 3415 IC50 < 280 nM T91442 CQ87XE 72187 IC50 = 5800 nM T91442 CU3P0Y 484047 IC50 = 70 nM T91442 C61SXL 492406 IC50 = 370 nM T91442 CZ1A8T 503580 IC50 = 770 nM T91442 C8F1DN 6482394 IC50 = 460 nM T36445 CJ73BT 45486346 Ki = 53 nM T36445 C9ETC4 45486354 Ki = 70 nM T36445 CVPG40 45486356 Ki = 3.65 nM T36445 CSQ2K4 45486357 Ki = 1.7 nM T36445 C0ET8W 137630787 Ki = 2 nM T36445 D0Y9PH 45486355 Ki = 0.75 nM T82467 CL80QG 11820 IC50 > 100000 nM T82467 C2IJU0 440987 IC50 > 1000000 nM T82467 CV56WH 1637655 IC50 = 23000 nM T82467 CM1AE9 3370466 IC50 = 7943.28 nM T82467 CGE54P 3573716 IC50 = 10000 nM T82467 CS9M8A 3577407 IC50 = 5011.87 nM T82467 CJ4U6Y 3589423 IC50 = 10000 nM T82467 C2U9DI 3657707 IC50 = 31622.78 nM T82467 CPN2V4 3673391 IC50 = 10000 nM T82467 C28EBX 4790771 IC50 > 100000 nM T82467 CXBG75 5125956 IC50 = 50118.72 nM T82467 CL91JP 9452375 IC50 = 79432.82 nM T82467 C1W7TE 16258532 IC50 = 1258.93 nM T82467 C25EUG 16272810 IC50 = 1258.93 nM T82467 CK2ES3 16313990 IC50 > 100000 nM T82467 CZ59FR 16316459 IC50 > 100000 nM T82467 CEN83U 16323492 IC50 = 12589.25 nM T82467 CM1R8O 16344932 IC50 > 100000 nM T82467 CO8M7K 17405877 IC50 = 31622.78 nM T82467 C9IP3Q 17446910 IC50 > 100000 nM T82467 CLP9S1 24687782 IC50 = 12589.25 nM T82467 CEL5F7 26851836 IC50 > 1000000 nM T82467 CG3PR6 52912222 IC50 > 31622.78 nM T82467 CF8B4E 60498769 IC50 > 100000 nM T82467 CHOS65 91820723 IC50 = 100000 nM T82467 C0TNJ7 91820724 IC50 = 12589.25 nM T82467 CAZ9M0 91826677 IC50 = 2511.89 nM T82467 CEN52P 91826678 IC50 = 1000 nM T82467 C3BR8O 118021718 IC50 > 80000 nM T82467 CC14FI 118933132 IC50 > 100000 nM T82467 CWC98G 121499171 IC50 = 2700 nM T82467 CO9J5W 122179607 IC50 = 15848.93 nM T82467 C3WOE8 122179608 IC50 = 50118.72 nM T82467 CW03JY 122179609 IC50 = 3981.07 nM T82467 CHNS18 122179610 IC50 = 1258.93 nM T82467 C2Q0OY 122179611 IC50 = 5011.87 nM T82467 C9GPL4 122179612 IC50 = 1995.26 nM T82467 CZX41C 122179613 IC50 = 1258.93 nM T82467 CJDK15 122179614 IC50 = 1584.89 nM T82467 CSF76G 122179615 IC50 = 794.33 nM T82467 CY7U0Z 122179616 IC50 = 1258.93 nM T82467 C1MV9L 122179617 IC50 = 1584.89 nM T82467 CJ81BV 122179618 IC50 = 3981.07 nM T82467 CZ69QO 122180530 IC50 > 100000 nM T82467 C7D5VP 122180531 IC50 > 100000 nM T82467 CRY84E 122180532 IC50 > 100000 nM T82467 C0J1AY 122180533 IC50 > 100000 nM T82467 CPIV02 122180534 IC50 > 100000 nM T82467 CC9XH7 122180535 IC50 > 100000 nM T82467 C0IWE1 122180536 IC50 = 501187.23 nM T82467 CEF19P 122180537 IC50 = 25118.86 nM T82467 C20LOD 122180538 IC50 = 63095.73 nM T82467 C73OMU 122180539 IC50 = 19952.62 nM T82467 CZSB51 122180540 IC50 = 31622.78 nM T82467 CJ4LO2 122180541 IC50 = 79432.82 nM T82467 C4TB0F 122180542 IC50 = 12589.25 nM T82467 CTXL15 122180543 IC50 = 15848.93 nM T82467 CUDY80 122180544 IC50 > 100000 nM T82467 C0SC2Y 122180545 IC50 > 100000 nM T82467 CR6T4G 122180546 IC50 = 50118.72 nM T82467 CHJG86 122180547 IC50 > 100000 nM T82467 CYZV97 122180548 IC50 > 100000 nM T82467 C0AIU8 122180549 IC50 = 50118.72 nM T82467 CPUS31 122180550 IC50 = 31622.78 nM T82467 CD62RB 122180551 IC50 = 39810.72 nM T82467 C8UCV9 122180552 IC50 = 7943.28 nM T82467 C72NLB 122180553 IC50 = 5011.87 nM T82467 CR0K5P 122180554 IC50 = 15848.93 nM T82467 CZ6L2N 122180555 IC50 = 6309.57 nM T82467 CKH49I 122180556 IC50 = 25118.86 nM T82467 CS4PD6 122180557 IC50 = 10000 nM T82467 CWC9I4 122180558 IC50 = 3162.28 nM T82467 CE7SL5 122180559 IC50 = 2511.89 nM T82467 CR6YD4 122180560 IC50 = 1258.93 nM T82467 C8HCK6 122180561 IC50 = 1258.93 nM T82467 CX9C6Y 122180562 IC50 = 3162.28 nM T82467 CPZ67Y 122180563 IC50 = 19952.62 nM T82467 CN1LE0 122180564 IC50 = 39810.72 nM T82467 CGLF82 122181547 IC50 = 199.53 nM T82467 CZGK74 122181548 IC50 = 125.89 nM T82467 C9P3GX 122181549 IC50 = 316.23 nM T82467 C3QJ5L 122181550 IC50 = 31.62 nM T82467 C3NC4V 122181552 IC50 = 125.89 nM T82467 C41ZXJ 122181555 IC50 = 199.53 nM T82467 C6I3VJ 122181557 IC50 = 39.81 nM T82467 C7CJR2 122181559 IC50 = 5011.87 nM T82467 CP5Z1C 122181560 IC50 = 1584.89 nM T82467 C61RTG 122181561 IC50 = 63095.73 nM T82467 CT62FG 122181571 IC50 = 79.43 nM T82467 C8F9VG 129196931 IC50 = 166 nM T82467 CO3A0E 134817551 IC50 = 251.19 nM T82467 CP4X5W 134817552 IC50 = 100 nM T82467 CA40QW 135535536 IC50 = 10000 nM T82467 CQT3A9 137636309 IC50 > 100000 nM T82467 CQ6XB7 139030526 IC50 = 316.23 nM T82467 CJ3FL8 145982835 IC50 = 251.19 nM T82467 CA2W8M 145984295 IC50 = 199.53 nM T82467 CE05ZV 145984432 IC50 = 25118.86 nM T82467 CV4GH7 145984467 IC50 = 251.19 nM T82467 CT6V0I 145985751 IC50 = 39.81 nM T82467 C0GHY5 145986052 IC50 = 125.89 nM T82467 CK98QJ 146035912 IC50 = 100 nM T82467 C2D1SB 155512075 IC50 = 1995.26 nM T82467 CD3LA9 155512613 IC50 = 1995.26 nM T82467 CE13CA 155515130 IC50 = 3981.07 nM T82467 CPM43N 155516232 IC50 > 100000 nM T82467 C23BXS 155517049 IC50 = 3162.28 nM T82467 C6Q3JK 155517968 IC50 = 1000 nM T82467 CFP24B 155518498 IC50 = 1995.26 nM T82467 CB49NL 155521254 IC50 = 63.1 nM T82467 CC30UG 155521851 IC50 = 1258.93 nM T82467 CL1P4M 155523233 IC50 = 1258.93 nM T82467 C1W8JL 155523577 IC50 = 50118.72 nM T82467 C2K9NI 155523694 IC50 = 2511.89 nM T82467 C0VS8H 155523850 IC50 = 1258.93 nM T82467 C3NYK0 155523937 IC50 = 1000 nM T82467 CW8O7G 155525483 IC50 = 794.33 nM T82467 CKR6V3 155528325 IC50 = 1584.89 nM T82467 COX8K5 155529510 IC50 = 1995.26 nM T82467 CVMC06 155529991 IC50 = 630.96 nM T82467 CL93CM 155530154 IC50 = 1000 nM T82467 CEI09V 155530332 IC50 = 251.19 nM T82467 CY7ST9 155530616 IC50 = 1000 nM T82467 CJ93LE 155531635 IC50 = 1995.26 nM T82467 C82UPM 155532741 IC50 = 3162.28 nM T82467 CAEQ29 155534550 IC50 = 1000 nM T82467 CY08SU 155535485 IC50 = 2511.89 nM T82467 CAL2G4 155538392 IC50 > 1000000 nM T82467 C9ISB5 155538742 IC50 = 2511.89 nM T82467 C1MQP2 155539283 IC50 = 1995.26 nM T82467 C45FSO 155539489 IC50 = 15848.93 nM T82467 CXTO91 155541586 IC50 = 2511.89 nM T82467 CSVH67 155541704 IC50 > 1000000 nM T82467 CNSP97 155542781 IC50 = 501.19 nM T82467 C6FHM8 155543582 IC50 = 630.96 nM T82467 CEA1C5 155545659 IC50 = 30 nM T82467 CM51BF 155546089 IC50 = 12589.25 nM T82467 CFTR89 155546746 IC50 = 1584.89 nM T82467 CRBT87 155547095 IC50 > 1000000 nM T82467 CQNO46 155548910 IC50 = 2511.89 nM T82467 C4VKR0 155551851 IC50 = 1258.93 nM T82467 C2FWB9 155551946 IC50 = 25.12 nM T82467 CT35SU 155553650 IC50 = 6309.57 nM T82467 C0SYN6 155554629 IC50 = 3162.28 nM T82467 CDO08V 155555578 IC50 = 3981.07 nM T82467 C12QHG 155555950 IC50 = 1584.89 nM T82467 C7S8GF 155556284 IC50 > 100000 nM T82467 C6N1CG 155557122 IC50 = 1000 nM T82467 CYM3K9 155557522 IC50 = 2511.89 nM T82467 CSGH17 155559412 IC50 = 1995.26 nM T82467 C1YWF9 155559659 IC50 > 1000000 nM T82467 C3IDR8 155559983 IC50 > 1000000 nM T82467 C5X6EL 155560182 IC50 = 251.19 nM T82467 CS1C5W 155560567 IC50 = 3162.28 nM T82467 C3UC7H 155560671 IC50 = 10000 nM T82467 C7EDG4 155564694 IC50 = 3162.28 nM T82467 C6MX5G 155564795 IC50 > 1000000 nM T82467 CXRJ70 155566441 IC50 = 1258.93 nM T82467 C2PIK0 155567275 IC50 = 1000 nM T82467 CM5FL1 155567534 IC50 = 2511.89 nM T82467 C7C9DH 155568184 IC50 = 6309.57 nM T82467 CZ2VN0 155569163 IC50 = 1258.93 nM T82467 D00XRH 91820725 IC50 = 1258.93 nM T82467 D0F5TZ 91827383 IC50 = 1258.93 nM T82467 D0O6XT 91827373 IC50 > 100000 nM T13260 D00AXJ 4189 IC50 = 600 nM T13260 D00ZFP 5870 Ki = 2500 nM T13260 D02STN 132971 IC50 > 5000 nM T13260 D04DJN 10635 Ki = 220 nM T13260 D06XMU 6013 Ki = 600 nM T13260 D07ABV 468595 IC50 = 8400 nM T13260 D09GOS 2812 IC50 = 1.8 nM T13260 D09LNI 3365 IC50 = 22000 nM T13260 D0B4IF 456201 IC50 = 951.48 nM T13260 D0C1WH 3902 Ki = 0.02 nM T13260 D0C7JF 13769 Ki = 35000 nM T13260 D0D2VS 60198 Ki = 10.2 nM T13260 D0G2MW 446284 IC50 = 53200 nM T13260 D0K8KX 5280343 IC50 = 12 nM T13260 D0M6DO 2145 IC50 = 5.2 nM T13260 D0Q5XX 445580 IC50 = 33200 nM T13260 D0W0BF 2187 Ki = 0.13 nM T13260 D0ZX1P 59693 Ki = 0.05 nM T13260 D03AJU 44139752 IC50 = 856 nM T13260 D05NJI 5287541 IC50 = 300 nM T13260 D08UGX 60652 IC50 = 44.67 nM T13260 D09NST 449459 IC50 = 530000 nM T13260 D0B4VE 10251 IC50 = 8000 nM T13260 D0G5CS 68071 IC50 = 900 nM T13260 D0L4FS 5280961 Ki = 100000 nM T13260 D0U3EP 445154 IC50 > 40 ug.mL-1 T13260 D0W4EB 10090750 IC50 = 6000 nM T13260 D0DK4I 4534 IC50 = 11 nM T13260 D03YPJ 5163 IC50 > 100000 nM T13260 D06JUR 56487 Ki = 1100 nM T13260 D09BKE 4553 IC50 = 680 nM T13260 D0C0JT 4495 IC50 = 27000 nM T13260 D0D3PF 6918191 IC50 = 1.38 nM T13260 D0SX7F 60876 Ki = 7.6 nM T13260 D0Y2OG 177865 IC50 = 0.5 nM T13260 C9LCD8 3823 IC50 = 60 nM T13260 C9NZY3 12452 Ki = 17 nM T13260 C2L1YD 22458 IC50 = 4110 nM T13260 CPY1G9 59694 Ki = 1.5 nM T13260 C87SRA 60796 IC50 = 1.4 nM T13260 CQ0IC4 63062 IC50 = 530000 nM T13260 CLJB07 65544 IC50 = 840 nM T13260 CHI68V 66425 Ki = 100 nM T13260 CG5ZC1 66842 Ki = 100 nM T13260 CMV4R6 67343 Ki = 100 nM T13260 C5JLH9 69088 IC50 > 125700 nM T13260 CRGU58 86488 IC50 = 19000 nM T13260 CR0XY7 88598 IC50 > 10000 nM T13260 CKN0O5 92267 IC50 > 16200 nM T13260 C2Q3LF 92775 IC50 = 9600 nM T13260 CEOP93 100332 IC50 > 40 ug.mL-1 T13260 C1D3WF 101928 IC50 = 1733 nM T13260 C56OAF 104880 Ki = 2.5 nM T13260 C1U3VY 124075 IC50 = 3920 nM T13260 CX30LQ 124600 IC50 = 4000 nM T13260 C64SKJ 125502 Ki = 60.9 nM T13260 CC1ES3 125503 Ki = 172 nM T13260 CPU8L1 125637 Ki = 18 nM T13260 CHWM72 125921 IC50 = 230 nM T13260 CV7MN1 126221 Ki = 17.6 nM T13260 CW45IU 126253 IC50 = 4600 nM T13260 C5E0PO 126735 IC50 = 61.66 nM T13260 CZW26T 128011 Ki = 5 nM T13260 C7CRO3 128300 Ki = 90 nM T13260 CV2KS6 129500 Ki = 5.8 nM T13260 C4UV3D 130636 Ki = 9.9 nM T13260 C7MK6N 131078 IC50 = 310 nM T13260 C9KN0L 131099 Ki = 170 nM T13260 C0JR2M 131426 Ki = 2220 nM T13260 CL0T6W 131798 IC50 = 5.754 nM T13260 C7N1EF 132907 Ki = 5 nM T13260 CL9ZS8 138203 IC50 = 11880 nM T13260 CF83MK 146141 Ki = 34 nM T13260 CPVI09 146142 Ki = 1 nM T13260 C1RTX5 146485 IC50 = 2700 nM T13260 C9H4TV 147045 Ki = 120 nM T13260 CWJ40O 151432 Ki = 120 nM T13260 C5AS9H 155976 IC50 > 40 ug.mL-1 T13260 C3Y7WX 158280 IC50 > 40 ug.mL-1 T13260 C9DTE4 160767 IC50 = 29000 nM T13260 CT5E1S 165184 IC50 > 50000 nM T13260 CYWS98 185848 IC50 > 40 ug.mL-1 T13260 CL5U9T 190972 Ki = 9.8 nM T13260 C0EOM6 193441 Ki = 1000 nM T13260 C1S9AI 196342 Ki = 15 nM T13260 CE4U0D 198531 IC50 > 50000 nM T13260 C36VAO 199390 IC50 > 50000 nM T13260 CU9BQ6 219377 IC50 = 46700 nM T13260 CAD54R 239595 IC50 = 250 nM T13260 C5WUK4 256446 IC50 = 4810 nM T13260 CQ6A8P 266151 IC50 = 800 nM T13260 COA9C7 280309 IC50 = 9000 nM T13260 C1C5TO 281901 Ki = 180 nM T13260 CS86KD 283391 IC50 = 20 nM T13260 CD8E9U 313177 IC50 = 37600 nM T13260 CE9R4U 316687 IC50 = 130 nM T13260 CNP1J9 334704 IC50 > 40 ug.mL-1 T13260 CU7L1E 343584 IC50 = 126000 nM T13260 CHL4T1 387487 IC50 = 95300 nM T13260 CA9B4J 390805 IC50 = 176000 nM T13260 C3AJN7 396930 IC50 = 100 nM T13260 CD2UN0 432882 IC50 = 11000 nM T13260 C7HME8 439246 IC50 = 2.9 nM T13260 CK2EB0 461948 IC50 = 6 nM T13260 CDM69B 484455 IC50 = 2160 nM T13260 CQ59RG 484458 IC50 = 580 nM T13260 CZO45T 484460 IC50 = 9230 nM T13260 CB2DY7 484461 IC50 = 1520 nM T13260 CS2RK5 484470 IC50 = 4000 nM T13260 CRED51 484475 IC50 = 3650 nM T13260 CLR9O8 492641 IC50 = 4590 nM T13260 CL21UY 508444 IC50 = 350 nM T13260 CQSN41 508446 IC50 = 300 nM T13260 CUWG73 508447 IC50 = 460 nM T13260 CQ4KL6 508448 IC50 = 2960 nM T13260 CS7DT2 508449 IC50 = 1510 nM T13260 C3GNC0 508450 IC50 = 1180 nM T13260 C7TVD8 508451 IC50 = 190 nM T13260 CW8JE3 508452 IC50 = 2200 nM T13260 CLAW60 508453 IC50 = 1530 nM T13260 C8L5OZ 510041 IC50 = 1240 nM T13260 CNB76G 510042 IC50 = 260 nM T13260 CH95MB 510043 IC50 = 1090 nM T13260 C9NGK0 510044 IC50 = 1370 nM T13260 CEZW17 510045 IC50 = 1040 nM T13260 CTLY25 510046 IC50 = 510 nM T13260 C7X6RO 510048 IC50 = 110 nM T13260 CX65UW 510049 IC50 = 1320 nM T13260 CXC2M7 510050 IC50 = 1680 nM T13260 CM23DG 510051 IC50 = 1000 nM T13260 C7TYH9 585624 IC50 = 3200 nM T13260 C5LJK2 591809 IC50 = 260 nM T13260 CI5FK2 591810 IC50 = 41000 nM T13260 C2QEF8 596715 IC50 > 50000 nM T13260 C3P1FA 606677 IC50 = 3050 nM T13260 CG72HV 622979 Ki = 58 nM T13260 CQ90BJ 623313 Ki = 140 nM T13260 CU4V9W 623696 Ki = 3000 nM T13260 CZ0AH3 638278 IC50 = 3800 nM T13260 CHV1X7 638701 IC50 = 3980 nM T13260 CM9IU5 641375 IC50 = 31100 nM T13260 CO28QU 641376 IC50 = 31100 nM T13260 CZ14PX 641378 IC50 > 40 ug.mL-1 T13260 CS2IQ3 715186 IC50 = 10600 nM T13260 CE4JQ8 782123 IC50 > 105800 nM T13260 C8EDM5 838923 IC50 = 39710 nM T13260 CFZ7C3 882273 IC50 = 5030 nM T13260 CP25US 1009065 IC50 = 50 nM T13260 CJQK73 1027647 IC50 = 529663443.9 nM T13260 CE9SH3 1291064 IC50 = 11600 nM T13260 C48SKB 1292107 IC50 = 2190 nM T13260 CEOM25 1294577 IC50 = 780 nM T13260 C6B9RE 1481465 IC50 = 22810 nM T13260 C1SH3T 1548910 IC50 > 50000 nM T13260 C7VE1Z 1548995 IC50 = 370000 nM T13260 CB93KS 1550302 IC50 = 9200 nM T13260 C3T8GZ 1831259 IC50 > 10000 nM T13260 CF18YS 2313447 IC50 = 1100 nM T13260 COYU39 2475352 IC50 = 200 nM T13260 CB4N3X 2725996 Ki = 234.3 nM T13260 C8SYF6 2725997 IC50 = 4 nM T13260 C68PUH 2725998 Ki = 63.38 nM T13260 CO84NG 2827372 IC50 = 16.5 nM T13260 CPXD41 2843385 IC50 = 1000 nM T13260 C3M7VX 2939932 IC50 = 10600 nM T13260 C8XJ1B 2992689 IC50 = 172 nM T13260 C3H1DE 2998104 IC50 = 1500 nM T13260 CUVM41 3035832 IC50 = 190 nM T13260 CZ1LD9 3298129 IC50 > 25000 nM T13260 C2SE4A 3346379 IC50 = 4300 nM T13260 C2OS4U 3361302 IC50 = 1100 nM T13260 CCD73S 3399276 IC50 = 3880 nM T13260 CBKQ75 3418244 IC50 = 370 nM T13260 C7O2MH 3943788 IC50 = 80 nM T13260 C40QVD 3964390 IC50 > 40 ug.mL-1 T13260 C7LX0V 4083407 IC50 = 59979107.63 nM T13260 C0WA7C 4103051 Ki = 830 nM T13260 CJ1U7P 4369413 IC50 = 100 nM T13260 CK17YZ 4369414 IC50 = 0.82 nM T13260 C1WIR4 4499193 IC50 > 31622.78 nM T13260 CXNH97 4993111 IC50 = 3670 nM T13260 C5OAR6 5121919 IC50 > 50000 nM T13260 CG0C4J 5281255 IC50 > 40 ug.mL-1 T13260 CM9Z0B 5312198 IC50 = 761 nM T13260 CF67ON 5314722 IC50 > 25000 nM T13260 CEW6B3 5315503 IC50 > 40 ug.mL-1 T13260 C3KDP7 5325467 IC50 = 16310 nM T13260 CW1UM5 5357488 IC50 > 351700 nM T13260 CBF75X 5376779 IC50 > 250000 nM T13260 CUV49J 5472143 IC50 = 5200 nM T13260 CR6N4L 5481966 IC50 > 40 ug.mL-1 T13260 C7VSM2 5702471 IC50 = 9332.54 nM T13260 CST49O 5702960 IC50 > 250000 nM T13260 C84XUK 6035693 IC50 = 5495.41 nM T13260 C3F7JB 6159604 IC50 = 12022.64 nM T13260 C1HZJ2 6438825 IC50 > 40 ug.mL-1 T13260 C2B1RH 6450879 IC50 > 40 ug.mL-1 T13260 CR8IB1 6457965 IC50 = 21700 nM T13260 C26KXD 6458748 IC50 = 2500 nM T13260 C39IEC 6461420 IC50 = 119 nM T13260 CP3O0B 6463551 IC50 = 61.6 nM T13260 CE93VI 6473542 IC50 = 100 nM T13260 C73LCV 6475119 IC50 = 42.7 ug.mL-1 T13260 C21BZK 6493479 IC50 = 63.7 nM T13260 CCO4Q3 6493484 IC50 = 440 nM T13260 CI13SQ 6523638 IC50 = 25000 nM T13260 C1JAT6 6539761 IC50 = 6580 nM T13260 CTE57C 6539762 IC50 = 3790 nM T13260 CF17BE 6539771 IC50 = 1130 nM T13260 CJ7RS8 6539772 IC50 = 4000 nM T13260 CP02JW 6539778 IC50 = 979489.99 nM T13260 CW1U8J 6539779 IC50 > 36000 nM T13260 CQD13Z 6539787 IC50 = 650 nM T13260 CQB1U5 6539798 IC50 = 800 nM T13260 C79FTC 6539799 IC50 = 1010 nM T13260 C5Z9KY 6539802 IC50 = 90 nM T13260 C7CAB8 6539809 IC50 > 36000 nM T13260 COU5D2 6539810 IC50 > 36000 nM T13260 CQ0HD5 6539812 IC50 = 720 nM T13260 CQ9XM0 6539813 IC50 = 1940 nM T13260 CF1R9J 6539815 IC50 > 36000 nM T13260 CMA37K 6539816 IC50 > 36000 nM T13260 CP4VI2 6540030 IC50 = 226 nM T13260 CR6LS8 6540031 IC50 = 190 nM T13260 CU3C1Y 6540034 IC50 = 125 nM T13260 CXEW82 6540035 IC50 = 119 nM T13260 CBKX32 6540037 IC50 = 120 nM T13260 C8MRI7 6540038 IC50 = 218 nM T13260 C8JXY1 6540039 IC50 = 20 nM T13260 CZK3T4 6540040 IC50 = 330 nM T13260 CDS26H 6540041 IC50 = 39 nM T13260 C2FRW5 6540044 IC50 = 970 nM T13260 C2JBQ1 6540045 IC50 = 810 nM T13260 CV0FA1 7330517 IC50 = 40950 nM T13260 CG9RF6 7515053 IC50 > 250000 nM T13260 C1DZ2H 7537616 IC50 = 150 nM T13260 C8VJ4X 8963350 IC50 > 50000 nM T13260 C0J1AS 9794431 IC50 = 10000 nM T13260 CS23XK 9797346 Ki = 10 nM T13260 C9QVL1 9816909 IC50 = 8900 nM T13260 CJ37SX 9818699 IC50 = 1.38 nM T13260 C2YB9F 9819524 IC50 = 12 nM T13260 CF7Z3J 9837392 IC50 = 2.9 nM T13260 C56CLB 9838063 IC50 = 680 nM T13260 CKJ1I6 9838340 IC50 = 580 nM T13260 CF3Z5V 9839853 Ki = 1.4 nM T13260 C35UMF 9890209 IC50 > 500000 nM T13260 CZ15MX 9908653 Ki = 36 nM T13260 CWL3O1 9926844 IC50 = 40000 nM T13260 C9Y3CA 9928113 IC50 = 12 nM T13260 CF24CV 9947889 Ki = 100 nM T13260 C0PHJ6 9948207 Ki = 70 nM T13260 C9BIH0 9948368 IC50 = 95.5 nM T13260 CZFV57 9949484 Ki = 1 nM T13260 CXH81D 9951467 IC50 = 0.12 nM T13260 CO1Z0A 9971194 IC50 = 5600 nM T13260 CBLP75 9972072 IC50 = 42.66 nM T13260 CDT6N2 9972577 IC50 = 8.8 nM T13260 C46LXP 9973019 Ki = 3.4 nM T13260 CB9DF4 9973046 IC50 = 20 nM T13260 C9JPT7 9974683 Ki = 1.4 nM T13260 CW1KO5 9976841 Ki = 36 nM T13260 C6W9NM 9978572 Ki = 16.5 nM T13260 C6Z0WQ 9991753 IC50 = 5000 nM T13260 CR16JI 9991838 IC50 = 530 nM T13260 CZV57I 9992344 IC50 = 6300 nM T13260 CQH4B7 9992433 IC50 = 14000 nM T13260 C2B4RF 9992450 IC50 = 4300 nM T13260 CVU3L0 9993026 IC50 = 3019.95 nM T13260 C85AUN 9998048 IC50 = 38.02 nM T13260 C0J8VR 10000064 IC50 = 78.5 nM T13260 C49HDL 10013868 IC50 = 170 nM T13260 C1FX2N 10014477 IC50 = 9300 nM T13260 C1KAV4 10015136 IC50 = 230 nM T13260 CPG39R 10018603 Ki = 3.4 nM T13260 C58EOH 10019839 IC50 = 130 nM T13260 CX7H2S 10020109 IC50 = 44 nM T13260 C0RP1F 10020714 IC50 = 44 nM T13260 CU12IF 10022210 IC50 = 130 nM T13260 CI7V2F 10023315 Ki = 36 nM T13260 C5PUD9 10026826 IC50 = 210 nM T13260 C5NAU2 10036028 IC50 = 600 nM T13260 C5Y0MK 10036693 IC50 = 380 nM T13260 CU7CI9 10042609 IC50 = 55 nM T13260 CV1K0G 10046399 IC50 = 51.8 nM T13260 C8MC0P 10051115 IC50 = 1650 nM T13260 C6W9NL 10060155 IC50 = 4200 nM T13260 C30LGM 10060824 IC50 = 3400 nM T13260 C64YSN 10064550 IC50 = 62 nM T13260 C9UMW8 10064832 IC50 = 600 nM T13260 C6Y1OT 10067777 Ki = 2.8 nM T13260 CI3S7F 10069029 IC50 = 220 nM T13260 CR13PX 10069113 Ki = 36 nM T13260 CX3FH6 10069477 Ki = 2.8 nM T13260 CR1V5S 10082665 IC50 = 93000 nM T13260 C64PHS 10083522 IC50 = 30 nM T13260 CR13LC 10084738 IC50 = 8700 nM T13260 CB65ED 10086187 Ki = 1.4 nM T13260 CL9X0W 10087126 Ki = 5000 nM T13260 C9YRP5 10087312 IC50 = 57 nM T13260 CPH49E 10087422 IC50 = 61.5 nM T13260 CD0MQ9 10088785 Ki = 1.4 nM T13260 CZB62D 10089657 Ki = 2.8 nM T13260 CNI2R6 10091150 IC50 = 102 nM T13260 C4JM1P 10104524 IC50 = 2400 nM T13260 C92KBY 10105573 IC50 > 19000 nM T13260 C7W5GI 10171354 IC50 = 14000 nM T13260 CD6JG2 10228895 IC50 = 500 nM T13260 CG2U1S 10242773 IC50 = 1000 nM T13260 CC08OX 10243987 IC50 = 590 nM T13260 CG24IZ 10247264 IC50 > 20000 nM T13260 CTK8F5 10248614 Ki = 9.3 nM T13260 C3YC9I 10263082 IC50 = 1900 nM T13260 C4CDG7 10264163 IC50 = 23000 nM T13260 CO2LT5 10286610 IC50 = 860 nM T13260 CD39LQ 10291777 IC50 = 100 nM T13260 CL6WE9 10295791 IC50 = 24000 nM T13260 C5LRW4 10298511 IC50 = 25100 nM T13260 CE2Z5S 10313881 IC50 = 41 nM T13260 C3PYH4 10317448 IC50 = 280 nM T13260 C6AOP4 10317522 IC50 = 530 nM T13260 CMO02D 10317756 Ki = 67000 nM T13260 C65BFK 10317931 IC50 = 400 nM T13260 C64YEQ 10318379 Ki = 9.8 nM T13260 CTUL01 10331100 IC50 = 185 nM T13260 CM81OX 10332392 IC50 = 3715.35 nM T13260 CZ4W0C 10332529 IC50 = 41 nM T13260 CQGS52 10334324 Ki = 1000 nM T13260 CQX4C8 10335739 Ki = 3.4 nM T13260 CT69PQ 10336071 IC50 = 100 nM T13260 C9RX2D 10338362 Ki = 9.3 nM T13260 CUDL75 10340374 Ki = 13.1 nM T13260 C0EO5N 10340839 Ki = 9.3 nM T13260 C07JGF 10355617 IC50 = 3300 nM T13260 CH5DS4 10358509 Ki = 5000 nM T13260 CWY9D0 10360147 Ki = 40 nM T13260 CELR79 10360875 IC50 = 63 nM T13260 CO69BI 10361506 IC50 = 49 nM T13260 CN7JK2 10368162 IC50 = 1650 nM T13260 CYNM04 10376335 IC50 = 260 nM T13260 CWY1X4 10379617 IC50 = 190 nM T13260 C5IZ0X 10380012 IC50 = 35000 nM T13260 CTX86G 10381606 IC50 = 233 nM T13260 COK7N8 10382166 IC50 = 1230 nM T13260 C06BMI 10384926 Ki = 13.1 nM T13260 C8CW6Y 10385742 Ki = 9.8 nM T13260 CP8G9A 10398594 IC50 = 13000 nM T13260 CXY9P7 10398686 IC50 = 1200 nM T13260 C1HZC5 10399349 IC50 = 240 nM T13260 CIJ01W 10400011 IC50 = 170 nM T13260 C3UN8Z 10400778 IC50 = 7900 nM T13260 CJ31WC 10403482 Ki = 42 nM T13260 C9LW2Z 10403903 IC50 = 49 nM T13260 CC5YT4 10404407 IC50 = 3000 nM T13260 CG7P5I 10404636 IC50 = 130 nM T13260 C9Q7CT 10407320 Ki = 36 nM T13260 C8KUR2 10421663 IC50 = 22000 nM T13260 C59NEQ 10426743 IC50 = 4300 nM T13260 CRV19P 10444266 IC50 = 1300 nM T13260 CR0O6C 10447478 IC50 = 20000 nM T13260 CTYP51 10448246 Ki = 5.1 nM T13260 CPAE70 10449017 IC50 = 1460 nM T13260 CUM3X2 10449331 IC50 = 2400 nM T13260 CQWX01 10450499 IC50 > 20000 nM T13260 C4L6ED 10450517 IC50 = 600 nM T13260 CM1IU9 10466775 IC50 = 6400 nM T13260 CT0H4G 10466776 IC50 = 750 nM T13260 C7TL6U 10467336 IC50 = 4786.3 nM T13260 C3YI0N 10467502 IC50 = 17000 nM T13260 C5DP9Z 10471817 IC50 = 10 nM T13260 CSM4H0 10472175 IC50 = 60 nM T13260 CIG25U 10474687 Ki = 10 nM T13260 C9W6YH 10488782 IC50 = 160 nM T13260 CYR2O4 10489655 IC50 = 680 nM T13260 CH7IA3 10489983 IC50 = 38000 nM T13260 CTW6A7 10494334 Ki = 17 nM T13260 CP8F4R 10495337 Ki = 4.7 nM T13260 CG0A6X 10513321 IC50 = 18000 nM T13260 CH2R0N 10513661 IC50 = 3900 nM T13260 C5RHY3 10538018 IC50 = 200 nM T13260 C7I6JP 10562688 IC50 = 239.88 nM T13260 CH8FS5 10565166 Ki = 3.1 nM T13260 C4L8OX 10566080 IC50 = 51000 nM T13260 C9PMK8 10566304 Ki = 12 nM T13260 C43DIK 10571994 Ki = 17 nM T13260 CN2RF5 10585362 IC50 > 250000 nM T13260 C7S5RV 10586086 IC50 = 220 nM T13260 CTI0R2 10587179 IC50 > 250000 nM T13260 CU5GI9 10594307 Ki = 5 nM T13260 C3RM0Y 10595083 Ki = 2.5 nM T13260 C3DH9W 10608774 IC50 = 920 nM T13260 CZ2H3N 10610950 IC50 > 250000 nM T13260 C02GMY 10617003 Ki = 2.5 nM T13260 CNR3V1 10618506 IC50 > 10000 nM T13260 C1F9IE 10636984 Ki = 5.3 nM T13260 C5TVC0 10637984 Ki = 12 nM T13260 CC39RI 10644237 Ki = 7 nM T13260 C04DNA 10656613 IC50 > 250000 nM T13260 C5ION6 10660701 IC50 = 3100 nM T13260 C9QN4J 10660816 IC50 = 36000 nM T13260 CJYQ87 10661641 Ki = 2.5 nM T13260 C8MOG9 10662151 Ki = 12 nM T13260 C8D0PV 10662758 Ki = 2.5 nM T13260 CUA2P0 10663766 Ki = 2.5 nM T13260 C8OUR1 10663913 Ki = 17 nM T13260 CPKA25 10665849 Ki = 17 nM T13260 CAYD96 10667894 Ki = 8.5 nM T13260 CP98RW 10680142 IC50 = 6000 nM T13260 CE12OS 10682353 IC50 = 24000 nM T13260 C0N2BV 10684551 IC50 = 9100 nM T13260 C01ZPW 10684552 IC50 = 10800 nM T13260 C1CGU5 10686589 Ki = 17 nM T13260 COB2W4 10690043 IC50 = 50 nM T13260 C0SIE5 10691220 Ki = 2.5 nM T13260 CMN02T 10708503 Ki = 1100 nM T13260 C1OME3 10710388 IC50 = 5200 nM T13260 CA13SW 10711620 IC50 = 549.54 nM T13260 CUQN16 10714213 IC50 > 10000 nM T13260 CO3JR0 10727176 IC50 = 51000 nM T13260 CBG72H 10729611 IC50 > 250000 nM T13260 CFE87L 10729612 IC50 = 27000 nM T13260 CYW4V9 10731755 IC50 > 10000 nM T13260 CKD29U 10738189 Ki = 9 nM T13260 CHL74J 10752290 IC50 = 103000 nM T13260 CU5W7P 10752634 IC50 = 350 nM T13260 CM3GX1 10753431 IC50 > 250000 nM T13260 C7U3ZR 10755577 IC50 = 4600 nM T13260 C4EXR1 10761806 IC50 = 1100 nM T13260 CZSA79 10774377 IC50 = 111000 nM T13260 CCD9R4 10774996 IC50 = 2400 nM T13260 C9GC0A 10775929 IC50 = 2600 nM T13260 CG27MD 10776192 IC50 > 250000 nM T13260 CNGQ30 10800145 IC50 = 1100 nM T13260 CJ5LW6 10806186 IC50 = 18100 nM T13260 CR25UM 10806331 Ki = 1100 nM T13260 C7P8IX 10810323 Ki = 10 nM T13260 CO53EU 10811011 Ki = 7 nM T13260 C0EAP2 10823139 IC50 = 700 nM T13260 C94PCN 10826001 IC50 = 8000 nM T13260 CN7I8H 10827014 IC50 = 16000 nM T13260 CZW6V4 10828130 IC50 = 2290.87 nM T13260 CM8WH3 10846478 IC50 = 3340 nM T13260 CU3I7B 10847200 IC50 = 440 nM T13260 CLZ5Q7 10853458 Ki = 37 nM T13260 C6RWM5 10854674 Ki = 17 nM T13260 C3UJ7E 10859502 Ki = 68 nM T13260 C26ARU 10859572 Ki = 22 nM T13260 CM5B1D 10883602 IC50 = 12 nM T13260 CVD0E9 10895435 IC50 > 40 ug.mL-1 T13260 CW9Z8X 10900865 IC50 > 40 ug.mL-1 T13260 CP85BH 10902291 Ki = 100 nM T13260 CWZC05 10903498 IC50 = 6.9 nM T13260 C59BGC 10904721 IC50 = 1.1 nM T13260 CXD1M3 10913975 IC50 > 40 ug.mL-1 T13260 C9UJN5 10914511 Ki = 60 nM T13260 CHX8K0 10927303 Ki = 70 nM T13260 CR6CX8 10957235 Ki = 170 nM T13260 C7QXL8 10958364 IC50 > 40 ug.mL-1 T13260 CX9N0T 10990534 IC50 > 40 ug.mL-1 T13260 C0VSL5 11001084 IC50 = 4500 nM T13260 CE3YX7 11015855 IC50 > 40 ug.mL-1 T13260 C04SCF 11023115 Ki = 110 nM T13260 CU5B1T 11033539 Ki = 58 nM T13260 CUQP81 11034900 Ki = 60 nM T13260 CZR21O 11066682 Ki = 250 nM T13260 CRE6W0 11078050 Ki = 90 nM T13260 CWR14N 11079165 IC50 = 39 nM T13260 C9IE5F 11085889 IC50 = 1600 nM T13260 CC2NG5 11109070 IC50 = 23 nM T13260 C52NIS 11140706 IC50 = 1800 nM T13260 CMB40V 11140772 IC50 = 2400 nM T13260 CDI1L7 11141249 Ki = 800 nM T13260 CZ31ND 11141567 IC50 = 5500 nM T13260 C5LS1V 11153057 Ki = 900 nM T13260 C63APE 11164320 IC50 = 610 nM T13260 C7TKN9 11164739 IC50 = 9200 nM T13260 CM59ZA 11176755 Ki = 1160 nM T13260 C1A9IY 11179136 IC50 = 530 nM T13260 C2KJ6H 11196148 IC50 = 168 nM T13260 CTA9B3 11197738 IC50 = 50 nM T13260 CFQ8X5 11213800 IC50 > 100000 nM T13260 C0IC8T 11218132 IC50 = 13900 nM T13260 CQ0IG4 11219074 IC50 = 3600 nM T13260 C1TP7W 11232831 IC50 = 150 nM T13260 CQGN76 11241635 IC50 = 31622.78 nM T13260 CR9UT3 11243132 IC50 = 100000 nM T13260 CC9X2S 11244229 IC50 > 100000 nM T13260 CD15BO 11244509 IC50 = 32 nM T13260 CFYD58 11246736 Ki = 1690 nM T13260 C8PJ7G 11265329 IC50 = 31622.78 nM T13260 C2A0GX 11276968 IC50 = 3380 nM T13260 C0V4IO 11288325 IC50 = 280 nM T13260 CR1JS5 11310894 IC50 = 9770 nM T13260 CRW74G 11322098 IC50 = 144 nM T13260 CI9H7S 11347268 Ki = 3.4 nM T13260 C8SK0O 11356920 IC50 = 1122.02 nM T13260 C9AO5H 11381850 IC50 > 50000 nM T13260 CXDT28 11392371 IC50 = 250 nM T13260 C5X7KI 11402766 IC50 = 26915.35 nM T13260 CH4VM5 11413971 IC50 = 2818.38 nM T13260 CX63YZ 11417114 IC50 = 3600 nM T13260 CF7J8A 11426612 IC50 = 5128.61 nM T13260 CAU8M0 11448232 IC50 = 2820 nM T13260 CO7U8R 11485667 IC50 > 100000 nM T13260 CA90VB 11493223 Ki = 100 nM T13260 CXP5I7 11493374 IC50 = 440 nM T13260 C8P4VL 11493892 IC50 = 960 nM T13260 CEFC74 11495013 IC50 = 12 nM T13260 CV02WR 11515409 IC50 = 1210 nM T13260 C3XAL1 11522408 IC50 = 15.3 nM T13260 CV58AY 11522728 IC50 = 470 nM T13260 CV3U7F 11530377 Ki = 100 nM T13260 CN4T0K 11544009 IC50 = 970 nM T13260 CDG7N4 11544414 IC50 = 110 nM T13260 CSW1P3 11551000 IC50 = 2810 nM T13260 CL5E7M 11558482 IC50 = 870 nM T13260 CAEQ30 11565696 IC50 = 300 nM T13260 CHJB42 11567631 IC50 = 0.92 nM T13260 CF51ZE 11568594 IC50 = 3.9 nM T13260 CX6OV1 11572776 Ki = 100 nM T13260 CVK75E 11572824 IC50 = 760 nM T13260 C5KNY1 11573432 IC50 = 630.96 nM T13260 COX19Z 11581191 IC50 = 176 nM T13260 C9IJ3T 11594132 IC50 = 1252 nM T13260 CBV48A 11595426 IC50 = 95.5 nM T13260 CKTA53 11603462 IC50 = 0.77 nM T13260 C3VHL8 11611589 IC50 = 99 nM T13260 CAM20K 11624089 Ki = 75 nM T13260 CB2L9J 11624690 IC50 = 160 nM T13260 C5Y6MN 11633212 IC50 = 25.5 nM T13260 C2UBZ0 11639518 IC50 = 290 nM T13260 C7SYX1 11644772 IC50 = 5870 nM T13260 C0ZD2V 11645369 IC50 = 230 nM T13260 C2WF8E 11653632 IC50 = 3960 nM T13260 C9QOK8 11654142 IC50 = 17.5 nM T13260 C1OU0F 11667385 IC50 = 2.291 nM T13260 CP6TI4 11681050 Ki = 147 nM T13260 CZA7U6 11687547 IC50 > 25000 nM T13260 CWH82Z 11696602 IC50 = 49 nM T13260 CZ50DQ 11708478 IC50 > 2000 nM T13260 C7WN6I 11716932 IC50 = 4490 nM T13260 CTHL93 11722357 Ki = 1.4 nM T13260 C59DIH 11723061 Ki = 4.9 nM T13260 CS4AR9 11723111 Ki = 3.4 nM T13260 CZH43C 11725276 IC50 = 1800 nM T13260 C0MD6A 11732219 IC50 = 2.3 nM T13260 CFB08O 11737365 IC50 = 0.06 nM T13260 CW2B3A 11738647 IC50 = 51 nM T13260 CD0KR5 11739060 IC50 = 107.15 nM T13260 CUTV09 11758702 IC50 > 16100 nM T13260 CLND03 11758964 IC50 = 150000 nM T13260 CG79IH 11760852 IC50 = 1800 nM T13260 CM2LK4 11774754 IC50 > 100000 nM T13260 CA7S0C 11779699 Ki = 5000 nM T13260 CIJQ20 11784241 IC50 > 50000 nM T13260 C83WAR 11792329 Ki = 2.5 nM T13260 C0LM8Q 11793414 Ki = 17 nM T13260 CIU5X2 11807837 Ki = 50 nM T13260 CZC18Q 11824496 IC50 = 1500 nM T13260 C3V9LP 11833981 IC50 = 420 nM T13260 C7W4TJ 11842924 IC50 = 910 nM T13260 CTCY19 11843079 IC50 = 2500 nM T13260 C81VMW 11843080 IC50 = 10000 nM T13260 C9YK3J 12137521 IC50 > 100000 nM T13260 CY0A2H 12846880 IC50 > 50000 nM T13260 CW7EC6 12854713 IC50 = 38300 nM T13260 CP94EZ 13257279 IC50 = 170000 nM T13260 CNKO41 13288738 IC50 = 54 nM T13260 C70ESC 13437151 IC50 > 50000 nM T13260 CW02LQ 13537950 IC50 = 245000 nM T13260 C90PFA 13537951 IC50 = 6000 nM T13260 CJ05FQ 13537952 IC50 = 2500 nM T13260 C6OQT1 13537953 IC50 = 3600 nM T13260 CAQK75 13537954 IC50 = 3200 nM T13260 CK6AZ4 13537955 IC50 = 330 nM T13260 C6RM8P 13537956 IC50 = 2400 nM T13260 C9XFJ0 13596071 Ki = 1750 nM T13260 C29SJW 13633181 Ki = 41 nM T13260 CY8V7Z 13633182 Ki = 36 nM T13260 C9LM0A 13633183 Ki = 73 nM T13260 CZP9U6 13633184 Ki = 36 nM T13260 CUX8Y6 13660214 IC50 > 300000 nM T13260 CJ41AQ 13660215 IC50 = 135000 nM T13260 CT0A6S 13660217 IC50 = 16000 nM T13260 CMR8V5 13660219 IC50 = 3000 nM T13260 C7YMZ1 13660220 IC50 = 3000 nM T13260 C9ZAK2 13660222 IC50 = 400 nM T13260 C6CVT0 13660223 IC50 = 1100 nM T13260 CL0B9C 13660224 IC50 = 600 nM T13260 CM26OE 13686727 IC50 = 1150 nM T13260 CB1XD6 13688211 IC50 = 3.2 nM T13260 C1F5IT 13688212 IC50 = 3.2 nM T13260 CA6Z5U 13688213 IC50 = 21 nM T13260 C0D4XQ 13688215 IC50 > 1000 nM T13260 CG0KB9 13688216 IC50 = 17.6 nM T13260 C3D8YA 13688218 IC50 = 14.3 nM T13260 CNF97R 13833941 IC50 = 880 nM T13260 C8LRB9 13900578 IC50 = 385000 nM T13260 CT1EY3 13900579 IC50 = 31000 nM T13260 C7IM0K 13900580 IC50 = 40000 nM T13260 CNC7F2 13900581 IC50 = 21000 nM T13260 CXLQ60 13900582 IC50 = 6600 nM T13260 C3HEP2 13900583 IC50 = 1500 nM T13260 C3DM0W 13900584 IC50 = 3000 nM T13260 C3TLJ9 13900585 IC50 = 10000 nM T13260 CS5G4U 13900586 IC50 = 30000 nM T13260 CG7O6E 13964844 Ki = 10000 nM T13260 C28GTK 13990942 Ki = 55 nM T13260 CS82TI 13990943 Ki = 53 nM T13260 CAY1C9 13991369 Ki = 100 nM T13260 C7LKS8 14055913 Ki = 690 nM T13260 CE6L1R 14055915 Ki = 260 nM T13260 CVU6D4 14068934 Ki = 1200 nM T13260 C27JCM 14068935 IC50 = 2500 nM T13260 C9X6BY 14068936 Ki = 50 nM T13260 CQO06Z 14068937 Ki = 1.5 nM T13260 CEK04X 14068938 Ki = 20 nM T13260 CY8M0H 14068939 IC50 = 4000 nM T13260 C7G8AL 14068940 IC50 = 200 nM T13260 C4WV0N 14068941 IC50 = 200 nM T13260 CYM3T7 14068942 IC50 = 2000 nM T13260 C8PIS0 14068943 IC50 = 7000 nM T13260 CNG31F 14068944 IC50 = 700 nM T13260 CDIY35 14077737 Ki = 45 nM T13260 C8GXN7 14097196 IC50 = 7.6 nM T13260 CLZ6B8 14097212 IC50 = 2 nM T13260 CN48CH 14097214 IC50 = 14.1 nM T13260 C0G6FZ 14131679 IC50 > 10000 nM T13260 CG3QI0 14166614 IC50 = 1180 nM T13260 C98EGQ 14196997 IC50 = 100 nM T13260 CL74NV 14213544 IC50 > 40 ug.mL-1 T13260 CI3FX8 14231148 IC50 = 47.86 nM T13260 CC8A0Q 14231150 IC50 = 10.96 nM T13260 CVG0J5 14231162 IC50 = 37.15 nM T13260 C67SBC 14231174 IC50 = 58.88 nM T13260 C58ATZ 14236566 IC50 > 40 ug.mL-1 T13260 CX17LO 14311671 Ki = 670 nM T13260 CDT9L8 14442755 Ki = 260 nM T13260 CJ2CW1 14442756 Ki = 103000 nM T13260 CJX8L5 14442758 Ki = 1198000 nM T13260 CL23QM 14442760 Ki = 130000 nM T13260 CY1G3T 14442762 Ki = 893000 nM T13260 CBI6E0 14442764 Ki = 13000 nM T13260 CI93VX 14442766 Ki = 8560 nM T13260 CKI1V2 14442768 Ki = 3980 nM T13260 C1LZV9 14442770 Ki = 45000 nM T13260 C2TWN4 14442772 Ki = 97000 nM T13260 CQ47RM 14542252 IC50 > 40 ug.mL-1 T13260 C91JNH 14607641 Ki = 100 nM T13260 CM4J5C 14670839 IC50 > 20000 nM T13260 C6CX1G 14732022 Ki = 46 nM T13260 C9OIP8 14777454 Ki = 12 nM T13260 CM52ZO 14777455 Ki = 12 nM T13260 CGE64N 14777478 Ki = 610 nM T13260 CB78FM 14852902 IC50 = 95.5 nM T13260 C3L8RM 14860771 Ki = 170 nM T13260 CYJU57 14860774 Ki = 289 nM T13260 CD6GC9 14860775 Ki = 170 nM T13260 C5EL2K 14860776 IC50 = 38000 nM T13260 CJ47KS 14860787 IC50 = 44000 nM T13260 C86IZO 14860791 IC50 = 100000 nM T13260 CUK4V7 14860794 Ki = 228 nM T13260 CUC7R6 14860795 Ki = 455 nM T13260 CT8X3G 14860799 Ki = 443 nM T13260 CQ2KA6 14860801 IC50 = 26000 nM T13260 CG41LP 14860811 Ki = 7750 nM T13260 C3TC1N 14872622 IC50 = 111 nM T13260 CIX71V 14872623 IC50 = 225 nM T13260 CLSM38 14872624 IC50 = 13 nM T13260 CN3O6Y 14872625 IC50 = 97 nM T13260 CY9G4S 14872626 IC50 = 240 nM T13260 CKW32M 14872634 IC50 = 2000 nM T13260 CK94GY 14872635 IC50 = 62 nM T13260 CD30OJ 14872636 IC50 = 31 nM T13260 C2OL5D 14872637 IC50 = 49 nM T13260 CLAX71 14890692 IC50 = 150 nM T13260 C62CXN 14890719 IC50 = 2100 nM T13260 C71PWS 14890720 IC50 = 13000 nM T13260 C92AQW 14927492 Ki = 1410 nM T13260 C92OWZ 14929519 IC50 > 98400 nM T13260 CP9F8I 14939800 IC50 = 17000 nM T13260 CS26UK 15068090 Ki = 926 nM T13260 C19BZH 15068091 Ki = 870 nM T13260 C3WMI4 15072946 IC50 = 6300 nM T13260 CRHI64 15072947 IC50 = 8912.51 nM T13260 CVU3M9 15072948 IC50 = 691.83 nM T13260 CD06BM 15072949 IC50 = 8600 nM T13260 CFM3T0 15072950 IC50 = 3000 nM T13260 C39GNY 15072951 IC50 = 2200 nM T13260 CBC15T 15072952 IC50 = 6200 nM T13260 CI2QF0 15072953 IC50 = 4900 nM T13260 CAM0B5 15079867 IC50 = 7.2 nM T13260 C69EXT 15079869 IC50 = 43.65 nM T13260 CB0HE6 15079883 IC50 = 95.5 nM T13260 C8KQE9 15180664 IC50 = 290 nM T13260 C3RQS5 15182462 IC50 = 3350 nM T13260 CJ09IM 15182464 IC50 = 69 nM T13260 C9KTC2 15182466 IC50 = 10000 nM T13260 C0H2MI 15182467 IC50 = 30.2 nM T13260 CQM9J1 15182468 IC50 = 370 nM T13260 C7D1CO 15182471 IC50 = 2800 nM T13260 CL7C3M 15182472 IC50 = 2818.38 nM T13260 C5YCE7 15182473 IC50 = 933.25 nM T13260 CB0K4F 15182475 IC50 = 330 nM T13260 C8LSJ6 15182477 IC50 = 66 nM T13260 C07YXF 15192231 IC50 = 96 nM T13260 CSR6T4 15250744 IC50 = 650 nM T13260 CL4E7S 15250885 Ki = 38 nM T13260 CRBA42 15250961 Ki = 100 nM T13260 CX03MI 15250962 Ki = 100 nM T13260 CG28BA 15341075 Ki = 6 nM T13260 CV05SR 15341076 Ki = 12 nM T13260 C30CFK 15383327 Ki = 58 nM T13260 CY5D3M 15485639 IC50 > 50000 nM T13260 C4E5CF 15516845 IC50 > 242400 nM T13260 C6W1EU 15541561 IC50 = 1700 nM T13260 C6FW0G 15658944 IC50 = 2700 nM T13260 CCEG42 15658945 IC50 = 800 nM T13260 C5FH9P 15658946 IC50 = 940 nM T13260 CS97IP 15658947 Ki = 36 nM T13260 CMZ08Y 15658949 Ki = 169 nM T13260 CXQG31 15680919 IC50 = 23000 nM T13260 C1OD2W 15680920 IC50 > 200000 nM T13260 CJ80RP 15680922 IC50 = 4100 nM T13260 C0NHV8 15680923 IC50 = 26000 nM T13260 CMD4C5 15703577 IC50 = 1200 nM T13260 C2CZB1 15710342 IC50 = 10000 nM T13260 CN4H6E 15754992 Ki = 2200 nM T13260 C2TB7G 15765776 IC50 = 42300 nM T13260 CZ32OY 15801213 Ki = 8.8 nM T13260 CV3N8J 15819093 Ki = 143 nM T13260 CTQK31 15926847 Ki = 1424 nM T13260 C7ZF5H 15926848 Ki = 1424 nM T13260 CK90YW 15926849 Ki = 61 nM T13260 CT7KD6 15926850 Ki = 60.9 nM T13260 C1T5KN 15926851 Ki = 174 nM T13260 CX7EL3 15926852 Ki = 60.9 nM T13260 CATK37 15926853 Ki = 94 nM T13260 C6FX8Y 15926855 Ki = 95 nM T13260 CYKA87 15926857 Ki = 88 nM T13260 CIN54V 15926859 Ki = 88 nM T13260 C31YEX 15949288 IC50 = 3000 nM T13260 CWIH26 16004744 IC50 = 180 nM T13260 CDO2P0 16051602 IC50 = 180 nM T13260 CA2MG0 16051603 IC50 = 700 nM T13260 CR0V1J 16051604 IC50 = 1100 nM T13260 CN05YL 16051605 IC50 = 1340 nM T13260 CBR91V 16051709 IC50 = 550 nM T13260 CI7AB0 16059386 IC50 = 20000 nM T13260 C4IX5G 16063410 IC50 = 12630 nM T13260 CAJ31C 16078976 IC50 = 3680 nM T13260 CU32JA 16114920 IC50 = 28300 nM T13260 C1WMH9 16124988 IC50 = 2170 nM T13260 C43QWJ 16124989 IC50 = 330 nM T13260 C0CA7G 16125055 IC50 = 2330 nM T13260 C9PM6N 16125056 IC50 = 7820 nM T13260 CG8R9J 16125059 IC50 = 580 nM T13260 CAT4J7 16125061 IC50 = 330 nM T13260 C30WQC 16125062 IC50 = 850 nM T13260 CY6T7B 16125116 IC50 = 230 nM T13260 CQI2W7 16125118 IC50 = 1170 nM T13260 C0A1WJ 16125119 IC50 = 370 nM T13260 CVG37K 16125176 IC50 = 810 nM T13260 CF93LW 16125180 IC50 = 400 nM T13260 C9JBA6 16125181 IC50 = 260 nM T13260 CDG07Z 16125182 IC50 = 490 nM T13260 CR9SW1 16125242 IC50 = 2680 nM T13260 C42SBM 16125249 IC50 = 1750 nM T13260 C4H7BV 16125314 IC50 = 7450 nM T13260 C9FQU1 16125315 IC50 = 5850 nM T13260 CXD90Z 16125316 IC50 = 5740 nM T13260 C8OYB6 16125317 IC50 = 470 nM T13260 CK1YQ5 16125318 IC50 = 1780 nM T13260 C3M9OJ 16125319 IC50 = 2400 nM T13260 C38VAJ 16125320 IC50 = 650 nM T13260 CU3X2I 16125321 IC50 = 520 nM T13260 CBL30A 16126879 IC50 = 70 nM T13260 C9BC0L 16732000 IC50 > 100000 nM T13260 C6G0AI 16737077 IC50 > 261500 nM T13260 C03XMV 16737078 IC50 > 261500 nM T13260 CI6AJ9 16737167 IC50 > 271400 nM T13260 CUB9P7 16737277 IC50 = 3670 nM T13260 C3IJ8X 16737837 IC50 = 13950 nM T13260 C6ITS8 16738014 IC50 = 4670 nM T13260 CZ7PO3 16738015 IC50 = 28650 nM T13260 C4VB7R 16738021 IC50 = 4080 nM T13260 C5B7NL 16738022 IC50 = 4750 nM T13260 CX5QL0 16738023 IC50 = 12100 nM T13260 CC9XH1 16738210 IC50 = 54670 nM T13260 CJNP76 16738212 IC50 = 82940 nM T13260 CEIO82 16738409 IC50 > 283750 nM T13260 CB79UM 16738411 IC50 = 7670 nM T13260 CCE5G1 16738412 IC50 = 25140 nM T13260 C8QEL7 16738421 IC50 > 295500 nM T13260 CF9ZR8 16738422 IC50 > 310200 nM T13260 CG3F9E 16747839 IC50 = 0.6 nM T13260 CUX1Q4 16747937 IC50 = 560 nM T13260 CN43EH 16747938 IC50 = 7.3 nM T13260 C19REJ 16747939 IC50 = 260 nM T13260 CFI2P7 16747940 IC50 = 5.3 nM T13260 CBZE53 16747941 IC50 = 31 nM T13260 C6RB8S 16747942 IC50 = 25.9 nM T13260 CC5OW7 16748063 IC50 = 17.7 nM T13260 C6H2YB 16748064 IC50 = 400 nM T13260 CVHS73 16748915 IC50 = 0.33 nM T13260 CFX0I7 16749017 IC50 = 1.5 nM T13260 C23CUO 16749018 IC50 = 2.8 nM T13260 CEB09A 16749022 IC50 = 27 nM T13260 C03MDH 16749112 IC50 = 0.88 nM T13260 C6L3DF 16749115 IC50 = 0.51 nM T13260 CS7G6V 16749118 IC50 = 7.6 nM T13260 C0C8HL 16749219 IC50 = 159 nM T13260 CZV59A 16749224 IC50 = 0.18 nM T13260 CNG1F9 16749332 IC50 = 0.5 nM T13260 CQNA43 16749333 IC50 = 1.2 nM T13260 CNHX39 16749336 IC50 = 0.4 nM T13260 CBU08D 16749337 IC50 = 42 nM T13260 C6U7AF 16749441 IC50 = 2.9 nM T13260 CG5KQ0 16749446 IC50 = 24 nM T13260 CC2YU9 17255947 IC50 = 28.7 nM T13260 CHUA83 17966236 Ki = 2400 nM T13260 CKQJ89 18599501 Ki = 8.2 nM T13260 C6WT3S 18628989 IC50 = 913 nM T13260 CZ7PK3 18632820 IC50 = 1000 nM T13260 CT85EY 18731901 IC50 > 50000 nM T13260 CK3SA5 19043020 IC50 = 288.4 nM T13260 C4YOJ7 19043038 IC50 = 147.91 nM T13260 CKX53Q 19043046 IC50 = 870.96 nM T13260 CNS3K1 20757276 IC50 = 750 nM T13260 CK87YW 20841680 Ki = 106 nM T13260 CSKO15 21044501 IC50 = 0.51 nM T13260 CVA07N 21044507 IC50 = 0.73 nM T13260 CA7ZH9 21121774 Ki = 610 nM T13260 C16NDX 21142052 IC50 > 12500 nM T13260 CWPF92 21278956 IC50 = 2300 nM T13260 C3K1MC 21682806 IC50 = 300 nM T13260 C9WKT3 21976841 IC50 = 2.8 nM T13260 CK2ZS8 21976856 IC50 = 43 nM T13260 CE7PI2 21976872 IC50 = 2.5 nM T13260 CN5FM4 21976888 IC50 = 15 nM T13260 C9CG8L 21976892 IC50 = 10 nM T13260 C6WC7P 21976903 IC50 = 2.9 nM T13260 C75VCH 21976905 IC50 = 178 nM T13260 CR9C7D 21976908 IC50 = 0.28 nM T13260 C1KU7Z 22278552 Ki = 150 nM T13260 CR73VN 22809920 Ki = 100 nM T13260 C25LBI 23220724 IC50 = 4580 nM T13260 CLV8H7 23365315 IC50 = 18.2 nM T13260 C9ALK0 23383196 IC50 = 270 nM T13260 CHL65N 23585513 IC50 = 14.4 nM T13260 CHW5O3 23585518 IC50 = 275 nM T13260 CMN52Q 23585571 IC50 = 0.2 nM T13260 CN3CK2 23585671 IC50 = 0.5 nM T13260 CWR42I 23585720 IC50 = 0.15 nM T13260 C43IUA 23585722 IC50 = 0.2 nM T13260 CVFG27 23585723 IC50 = 0.1 nM T13260 CVJ95M 23585770 IC50 = 6 nM T13260 C30WOI 23585773 IC50 = 74 nM T13260 C5VWK3 23644932 Ki = 1820 nM T13260 CT8BJ4 23644933 Ki = 250 nM T13260 C6D9MC 23644934 Ki = 4400 nM T13260 COB81D 23644935 IC50 = 18000 nM T13260 C91ZAQ 23644936 IC50 > 50000 nM T13260 CWX70I 23644937 IC50 > 50000 nM T13260 C2I1BV 23644938 IC50 > 50000 nM T13260 C13NZL 23644951 IC50 = 85 nM T13260 CKBT84 23644968 Ki = 54 nM T13260 CC7FB8 23644969 Ki = 19 nM T13260 CJ3FX4 23644970 Ki = 22 nM T13260 C40DSL 23644971 Ki = 16 nM T13260 C8LJ4B 23644972 Ki = 11 nM T13260 C38VLD 23644973 Ki = 25 nM T13260 CNQ12D 23644974 Ki = 20 nM T13260 CR8VS6 23644975 Ki = 43 nM T13260 CF47DK 23644976 Ki = 4.7 nM T13260 CH5L6T 23644977 Ki = 7 nM T13260 CY1EL0 23644978 Ki = 14 nM T13260 C20LOE 23644979 Ki = 5 nM T13260 CDZN28 23644980 Ki = 8 nM T13260 CBVS04 23644981 Ki = 7.8 nM T13260 CO26RY 23644982 IC50 = 0.037 nM T13260 C4BPW5 23644983 IC50 = 0.11 nM T13260 CYV81F 23644984 IC50 = 0.23 nM T13260 CGF0J4 23644985 IC50 = 9 nM T13260 CVX82D 23644986 IC50 > 50 nM T13260 CG98LY 23644987 IC50 = 0.049 nM T13260 C9JD7L 23644988 IC50 = 0.32 nM T13260 C9JHP1 23644989 IC50 = 0.44 nM T13260 C7ZTD4 23644990 IC50 = 12 nM T13260 COF70P 23644991 IC50 > 50 nM T13260 CYG5P8 23644992 IC50 = 0.19 nM T13260 C74ILW 23644993 IC50 = 0.16 nM T13260 C5T6NR 23644994 IC50 = 0.12 nM T13260 C6FK7A 23644995 IC50 = 0.05 nM T13260 CIN07U 23644996 IC50 = 0.26 nM T13260 C8NY5J 23644997 IC50 = 0.13 nM T13260 C6EZ5V 23644998 Ki = 0.38 nM T13260 C0KZA5 23644999 Ki = 0.18 nM T13260 CKH5D2 23645000 Ki = 2.9 nM T13260 C27FSX 23645001 Ki = 44 nM T13260 CIQ42N 23645002 IC50 > 50 nM T13260 CX8Q9F 23645003 Ki = 0.14 nM T13260 C50OAY 23645004 Ki = 0.34 nM T13260 C5I6RZ 23645005 Ki = 5.5 nM T13260 C6PFS4 23645006 IC50 > 50 nM T13260 CIKQ38 23645007 IC50 > 50 nM T13260 C2DK6T 23645008 Ki = 0.045 nM T13260 CM2JR9 23645024 IC50 = 7400 nM T13260 C0HD7V 23645025 IC50 = 22 nM T13260 C73XCN 23645026 IC50 = 870 nM T13260 CTU28I 23645027 IC50 > 10000 nM T13260 CTUW15 23645028 IC50 > 10000 nM T13260 CL35CQ 23645029 IC50 = 10000 nM T13260 C2P7DG 23645030 IC50 > 10000 nM T13260 C89VHK 23645031 IC50 > 10000 nM T13260 CGKW86 23645032 IC50 > 1000 nM T13260 C2I9XH 23645033 IC50 = 400 nM T13260 C3J6KZ 23645034 IC50 > 10000 nM T13260 CEM21C 23645035 IC50 > 1000 nM T13260 CQ1KF8 23645036 IC50 > 1000 nM T13260 C1IT7Q 23645037 IC50 > 1000 nM T13260 CM81SC 23645038 IC50 > 1000 nM T13260 CA7DX4 23645039 IC50 > 1000 nM T13260 C1CQ4N 23645040 IC50 = 1000 nM T13260 CJV60Q 23645041 IC50 = 570 nM T13260 CQH8D4 23645042 IC50 = 270 nM T13260 C9L5EJ 23645043 IC50 = 50 nM T13260 C1X5NC 23645044 IC50 > 1000 nM T13260 CA76DP 23645045 IC50 > 1000 nM T13260 CLK43G 23645046 IC50 > 1000 nM T13260 C74MFK 23645047 IC50 = 330 nM T13260 CF48RD 23645048 IC50 = 50 nM T13260 C3A5VO 23645049 IC50 > 1000 nM T13260 CS2T8L 23645050 IC50 > 1000 nM T13260 CB24PD 23645051 IC50 > 1000 nM T13260 CLCA31 24204030 IC50 = 3100 nM T13260 CQ41JU 24204037 IC50 = 2400 nM T13260 CPJ8Z9 24205803 IC50 = 4400 nM T13260 CRH52Y 24205804 IC50 = 9100 nM T13260 C2PYN1 24420563 IC50 = 160 nM T13260 CP1YO7 24424201 IC50 = 800 nM T13260 CGVM50 24431784 IC50 > 50000 nM T13260 C6D2NZ 24692916 IC50 = 3715.35 nM T13260 CBU73T 24806841 IC50 > 25000 nM T13260 CA0YQ2 24806842 IC50 > 25000 nM T13260 CC92RE 24806843 IC50 > 25000 nM T13260 C17MET 24807041 IC50 > 25000 nM T13260 C9CMI7 24807042 IC50 > 25000 nM T13260 CZ6I0R 24807043 IC50 > 25000 nM T13260 CMY75P 24807044 IC50 > 25000 nM T13260 CJO96W 24807045 IC50 > 25000 nM T13260 CS8GB3 24807046 IC50 = 2170 nM T13260 C2B4HN 24807239 IC50 = 17370 nM T13260 C39TNQ 24807240 IC50 = 1100 nM T13260 C3PRI8 24807241 IC50 = 16670 nM T13260 CM4P0V 24807242 IC50 = 1770 nM T13260 CS01MP 24807243 IC50 = 250 nM T13260 C3BSZ8 24807244 IC50 = 690 nM T13260 CNTI27 24807245 IC50 = 690 nM T13260 C18DIO 24807434 IC50 = 440 nM T13260 C6CA8F 24807435 IC50 = 1070 nM T13260 C8NR1Y 24807436 IC50 = 120 nM T13260 CC73NY 24873506 IC50 = 1370 nM T13260 CAX9V3 24873507 IC50 = 1540 nM T13260 CS2IG5 24873508 IC50 = 610 nM T13260 C5TA7V 24873509 IC50 = 630 nM T13260 CW3C5U 24896569 IC50 = 38 nM T13260 CS5H2A 24896701 IC50 > 15300 nM T13260 CBZ10U 24901645 IC50 = 13 nM T13260 CY27CS 24901646 IC50 = 12 nM T13260 CD9IV7 24901647 IC50 = 3 nM T13260 CMFU23 24901648 IC50 = 3.2 nM T13260 CTJ76G 24901649 IC50 = 14.3 nM T13260 CJ7R6C 24901650 IC50 = 2457 nM T13260 CVS08H 24901651 IC50 = 169 nM T13260 C2H8EA 24901652 IC50 = 215 nM T13260 CUF1O4 24901653 IC50 = 5.5 nM T13260 C9C0AB 24901654 IC50 = 1.8 nM T13260 CEB6G1 24901655 IC50 = 0.6 nM T13260 CE5QO1 24901656 IC50 = 3.4 nM T13260 C23PCS 25022806 IC50 = 13.7 nM T13260 CF02OB 25071641 IC50 = 11.5 nM T13260 CMXL59 25111668 Ki = 2100 nM T13260 C35FYQ 25111796 IC50 > 500000 nM T13260 C8J2AP 25111799 IC50 > 500000 nM T13260 C06ECA 25111909 Ki = 1530 nM T13260 CON29S 25141424 IC50 = 0.45 nM T13260 CZX08M 25142015 Ki = 13 nM T13260 CV2DP9 25180002 IC50 = 6500 nM T13260 C0XHA2 25180109 IC50 = 426 nM T13260 CS8YW6 25227426 IC50 = 33000 nM T13260 CC1S3T 25256841 IC50 = 24400 nM T13260 CA4G8Y 42597583 IC50 = 13 nM T13260 C5N9MC 42611455 IC50 = 5300 nM T13260 C93BZJ 42618027 IC50 = 1250 nM T13260 C4YXR5 42618028 IC50 = 31500 nM T13260 CVLR83 42618034 IC50 = 5680 nM T13260 CUWO14 42618035 IC50 = 760 nM T13260 CZW8L2 43137984 IC50 = 289 nM T13260 CCZY29 44266320 IC50 = 620 nM T13260 C1BGQ4 44266331 IC50 = 1600 nM T13260 CEHD28 44266353 IC50 = 800 nM T13260 C79VFZ 44275189 Ki = 12 nM T13260 CQ31TG 44275201 Ki = 22 nM T13260 C83QEP 44275202 Ki = 6.7 nM T13260 CDK2T1 44275250 Ki = 5.1 nM T13260 CJ48ZL 44275251 Ki = 63 nM T13260 C78OQW 44275252 Ki = 31 nM T13260 CG4FB5 44275253 Ki = 10 nM T13260 C0OE3W 44275268 Ki = 21 nM T13260 CZ9K6I 44275269 Ki = 11 nM T13260 CP29RM 44275270 Ki = 37 nM T13260 CP2QV1 44275283 Ki = 5.6 nM T13260 C1A6OS 44275328 Ki = 4.7 nM T13260 CLN69H 44275329 Ki = 62 nM T13260 C1LQC6 44275331 Ki = 1.4 nM T13260 CZWI57 44275351 Ki = 8.8 nM T13260 C9R1OJ 44275355 Ki = 4.6 nM T13260 CC30JG 44276238 IC50 = 777000 nM T13260 CN9W6A 44276773 Ki = 75 nM T13260 C7GMW1 44277065 Ki = 1 nM T13260 C76XWA 44277083 Ki = 7 nM T13260 C3SU7M 44286352 IC50 = 170 nM T13260 CH4TJ0 44286353 IC50 = 2900 nM T13260 C74AKY 44286427 IC50 = 200 nM T13260 C0KVR6 44286475 IC50 = 70 nM T13260 C4WE8P 44286839 IC50 = 110 nM T13260 C2T1CJ 44286840 IC50 = 90 nM T13260 CZO6F2 44287464 Ki = 30 nM T13260 C8D9XI 44287465 Ki = 27 nM T13260 CK76RT 44287659 IC50 = 4400 nM T13260 C08POV 44287660 IC50 = 10000 nM T13260 CMA78S 44287741 IC50 = 4400 nM T13260 CGUX54 44287754 IC50 = 1200 nM T13260 CNF17L 44287801 Ki = 30 nM T13260 C5F6MV 44294033 Ki = 63 nM T13260 CHNJ98 44294100 Ki = 27 nM T13260 C7T9RN 44294311 Ki = 926 nM T13260 C5U1JS 44294312 Ki = 870 nM T13260 CMW32B 44294314 Ki = 11 nM T13260 C5JHW7 44294332 Ki = 190 nM T13260 C4TY5K 44306234 IC50 = 200 nM T13260 CCE7A4 44306491 IC50 = 52020 nM T13260 CUQ6L9 44306493 IC50 = 2170 nM T13260 CGU34E 44306494 IC50 = 3000 nM T13260 C9GRJ2 44306526 IC50 = 590 nM T13260 CN34EP 44306915 IC50 = 190 nM T13260 C8RQ5W 44306929 IC50 = 880 nM T13260 C80ZJS 44307719 Ki = 47 nM T13260 C76BWU 44307720 Ki = 28 nM T13260 CM52NG 44307837 Ki = 100 nM T13260 CF1K2N 44310044 Ki = 3000 nM T13260 CB30FN 44310045 Ki = 1800 nM T13260 C0QZ5L 44310046 Ki = 7000 nM T13260 C3QWV2 44310077 Ki = 13000 nM T13260 C32AUZ 44310078 Ki = 2000 nM T13260 CLJ45R 44310148 Ki = 1400 nM T13260 CEOU45 44310393 Ki = 5500 nM T13260 CZMQ71 44310410 Ki = 11000 nM T13260 CKNF03 44310411 Ki = 45000 nM T13260 C6X7WP 44310412 Ki = 9800 nM T13260 C90SJZ 44310767 Ki = 5300 nM T13260 C8W3VA 44310768 Ki = 11000 nM T13260 CO2SE0 44323417 IC50 = 3200 nM T13260 CRW0C1 44323482 IC50 = 2400 nM T13260 C0FAY8 44323523 IC50 = 2500 nM T13260 CRG1T9 44323592 IC50 = 31000 nM T13260 CQM56K 44323610 IC50 = 10000 nM T13260 C63FUL 44323664 IC50 = 3000 nM T13260 CVF86M 44323741 IC50 = 245000 nM T13260 CZIS73 44323756 IC50 = 21000 nM T13260 C0J6ZI 44323759 IC50 = 3600 nM T13260 CQC0G4 44323760 IC50 = 30000 nM T13260 CADY94 44323768 IC50 = 800 nM T13260 CGK6B2 44323782 IC50 = 1500 nM T13260 CQT35R 44323783 IC50 = 6600 nM T13260 CR5S8Z 44323807 IC50 = 40000 nM T13260 C87RGX 44323808 IC50 = 385000 nM T13260 CY1OB4 44323813 IC50 = 4000 nM T13260 CI0H9D 44323814 IC50 = 6000 nM T13260 CLE87R 44328597 Ki = 18.9 nM T13260 CX8DV2 44328668 Ki = 13.1 nM T13260 CXS8N4 44330891 Ki = 25000 nM T13260 C38YFI 44330892 Ki = 1100 nM T13260 C09VTC 44330997 Ki = 12 nM T13260 CFW8Q5 44330998 Ki = 3000 nM T13260 C5CF2O 44331012 Ki = 4.7 nM T13260 CQ85VL 44331071 Ki = 1 nM T13260 CL1YN0 44331102 Ki = 35000 nM T13260 CJIW38 44331119 Ki = 56 nM T13260 CHY39A 44331123 Ki = 1.3 nM T13260 C2MZO4 44331205 Ki = 2.3 nM T13260 CZHI57 44331221 Ki = 3 nM T13260 CXY2W3 44331222 Ki = 9 nM T13260 C28YNW 44331250 Ki = 33000 nM T13260 CR1YC8 44331322 IC50 = 30 nM T13260 CQR2U5 44333942 IC50 = 340 nM T13260 CL4Q0F 44333943 IC50 = 97 nM T13260 CX6Q1N 44334361 IC50 = 89 nM T13260 CB2D4V 44334394 IC50 = 9700 nM T13260 CSO4C8 44334411 IC50 = 11800 nM T13260 CCZ60G 44334579 IC50 = 310 nM T13260 CBZV02 44334580 IC50 = 120 nM T13260 CSR90W 44334594 IC50 = 2000 nM T13260 C8GAF6 44334595 IC50 = 3200 nM T13260 CIB4F8 44339828 Ki = 37 nM T13260 CS2F5B 44340058 Ki = 10 nM T13260 C7PT2A 44340059 Ki = 47.6 nM T13260 C9YAC2 44340330 Ki = 65.8 nM T13260 C0SC3B 44341451 IC50 = 5400 nM T13260 CAD1S9 44341468 IC50 = 238 nM T13260 CKE5L8 44353429 IC50 = 236 nM T13260 CYO3B6 44353430 IC50 = 245 nM T13260 C0UDL7 44353435 IC50 = 342 nM T13260 C3XP8T 44353437 IC50 = 950 nM T13260 C0KIV8 44353626 IC50 = 800 nM T13260 CME45Q 44353627 IC50 = 658 nM T13260 CX43HZ 44353643 IC50 = 490 nM T13260 CQ5UK0 44354378 IC50 = 530 nM T13260 CO8XJ3 44354706 IC50 = 120 nM T13260 C7YDP6 44354757 IC50 = 1320 nM T13260 C1W6IR 44354758 IC50 = 3960 nM T13260 C4AXM5 44354773 IC50 = 440 nM T13260 CZN1X8 44354907 IC50 = 30000 nM T13260 CN8M5U 44354930 IC50 = 5600 nM T13260 CCA28Y 44354942 IC50 = 55000 nM T13260 CNRO38 44354943 IC50 = 3850 nM T13260 CQIP34 44354944 IC50 = 80500 nM T13260 CO1W4F 44355172 IC50 = 8900 nM T13260 CX2R3P 44355187 IC50 > 20000 nM T13260 CCF7G1 44355188 IC50 = 1700 nM T13260 C64IWU 44358640 IC50 = 7100 nM T13260 CR5M1D 44369877 Ki = 18 nM T13260 C3BDK1 44369898 Ki = 65 nM T13260 CKNO08 44369927 Ki = 59 nM T13260 CL19DY 44376315 IC50 = 92.9 nM T13260 CZE46J 44378054 IC50 = 42 nM T13260 C1I0NW 44381001 IC50 > 250000 nM T13260 CDTS58 44387709 IC50 = 15 nM T13260 CUNZ83 44394828 IC50 = 1400 nM T13260 C8I1AE 44394829 IC50 = 31600 nM T13260 C2TLS9 44404116 Ki = 50 nM T13260 CLV8R2 44408288 IC50 = 29.7 nM T13260 C9DS0J 44408292 IC50 = 26.3 nM T13260 CTD91Q 44408293 IC50 = 23.7 nM T13260 C5X7TN 44408294 IC50 = 19.3 nM T13260 CIBP08 44421541 IC50 = 57.54 nM T13260 C0WU4A 44421546 IC50 = 93.33 nM T13260 CCIE32 44421551 IC50 = 3715.35 nM T13260 C9A6IF 44421559 IC50 = 47.86 nM T13260 C5FO6U 44424773 IC50 > 310170 nM T13260 C6BE0T 44456226 IC50 > 5000 nM T13260 CY7OD4 44461241 IC50 > 50000 nM T13260 C4BAS8 44462074 Ki = 228 nM T13260 C9BE8F 44462253 Ki = 455 nM T13260 C92QWL 44521066 IC50 = 0.12 nM T13260 CG16BM 44554135 IC50 = 11500 nM T13260 C47OVI 44562528 IC50 > 500000 nM T13260 CY42QT 44562549 IC50 > 500000 nM T13260 CP3T7B 44567161 IC50 > 40 ug.mL-1 T13260 C90PBX 44567164 IC50 > 40 ug.mL-1 T13260 C49DYC 44567218 IC50 = 7500 nM T13260 CO63LK 44569291 IC50 = 2.3 nM T13260 CNZV98 44577912 IC50 = 93.8 nM T13260 CRP8A7 44577913 IC50 = 18.7 nM T13260 CW8XY2 44577949 IC50 = 1620 nM T13260 C5CSL8 44578878 IC50 = 17300 nM T13260 C2ZWD9 44578879 IC50 = 5060 nM T13260 C4F2AM 44578880 IC50 = 1040 nM T13260 C1AT7Y 44578921 IC50 = 1060 nM T13260 C60AKC 44579025 IC50 = 320 nM T13260 C50KAN 44579026 IC50 = 9960 nM T13260 CJQ67H 44579027 IC50 = 2490 nM T13260 CS4JR7 44579028 IC50 = 1070 nM T13260 CHWK61 44579029 IC50 = 870 nM T13260 C8QW4K 44579570 IC50 = 13040 nM T13260 CP53WC 44580785 IC50 = 17000 nM T13260 CGBT61 45028483 IC50 > 10000 nM T13260 CVO41F 45140953 IC50 = 2 nM T13260 CRZ6N5 45140954 IC50 = 0.5 nM T13260 C01WQZ 45141152 IC50 = 2.4 nM T13260 CT5CR6 45141153 IC50 = 0.22 nM T13260 CC3FT1 45141154 IC50 = 0.35 nM T13260 C8PB0I 45141156 IC50 = 146 nM T13260 CL2Y7U 45141157 IC50 = 29.3 nM T13260 CH1LB7 45141158 IC50 = 19 nM T13260 CDE83B 45141365 IC50 = 52 nM T13260 CGA6Y4 45141366 IC50 = 112 nM T13260 CCIP58 45141367 IC50 = 280 nM T13260 C2S5QX 45141368 IC50 = 24 nM T13260 C2YJ8N 45141369 IC50 = 80 nM T13260 CO4UA1 45141370 IC50 = 920 nM T13260 C5CB0P 45141371 IC50 = 284 nM T13260 CTN65F 45141372 IC50 = 380 nM T13260 CGK5O7 45141601 IC50 = 571 nM T13260 C68SZB 45141602 IC50 = 0.8 nM T13260 C0C3AW 45141603 IC50 = 1.9 nM T13260 C0U7CG 45141604 IC50 = 0.3 nM T13260 CQ4JE3 45378299 IC50 = 97000 nM T13260 CUR6C8 45378303 IC50 = 5100 nM T13260 CY2SV8 45379302 IC50 = 44000 nM T13260 CSE09V 46177290 IC50 = 12100 nM T13260 C4XCR3 46177291 IC50 = 12100 nM T13260 C4S2AI 46198256 Ki = 16.1 nM T13260 CT07FB 46204132 IC50 = 6400 nM T13260 CN47GA 46228644 IC50 = 4.6 nM T13260 C6AMH8 46228668 IC50 = 1.7 nM T13260 CLD4Z5 46228698 IC50 = 0.22 nM T13260 CZH36E 46834487 IC50 > 50000 nM T13260 CUV83E 46854605 IC50 = 12000 nM T13260 CIA08B 46854608 IC50 = 9500 nM T13260 CWJ3F1 46854758 IC50 = 5060 nM T13260 CKRQ67 46854759 IC50 = 49500 nM T13260 CZ1YJ0 46854760 IC50 = 48700 nM T13260 CINV65 46867541 IC50 = 101 nM T13260 CL06TP 46887017 IC50 = 17.2 nM T13260 C0KFI6 46887054 IC50 = 17.2 nM T13260 C6R1HA 46887055 IC50 = 6 nM T13260 CD65CW 46887468 IC50 = 71.8 nM T13260 CM0EK7 46887507 IC50 = 200 nM T13260 CGBE96 46887549 IC50 = 210 nM T13260 C74CER 46887577 IC50 = 3.5 nM T13260 C2OMW7 46895138 IC50 = 12000 nM T13260 CYEA34 46913124 IC50 = 70 nM T13260 C5JR7T 46913125 IC50 = 36 nM T13260 CN1CV7 46939057 Ki = 97 nM T13260 CP8HY2 46939058 Ki = 27 nM T13260 CD67MH 46939156 Ki = 23 nM T13260 C1MFE9 46939157 Ki = 75 nM T13260 C0K8YL 46939158 Ki = 39 nM T13260 CX7B9G 46939159 Ki = 30 nM T13260 CL37EV 46939160 Ki = 56 nM T13260 C9CQU0 46953209 IC50 = 59.2 nM T13260 CUQ0Z7 46957695 IC50 = 13200 nM T13260 CU0KW6 46958302 IC50 = 991 nM T13260 CHN2P9 46960541 IC50 = 34.5 nM T13260 CR3OI4 46960542 IC50 = 46.7 nM T13260 CW3V2P 46962897 IC50 = 499 nM T13260 CQ0XE9 46964149 IC50 = 10600 nM T13260 CL0F1J 46964152 IC50 > 25000 nM T13260 CV3UT0 46967737 IC50 = 3100 nM T13260 CBAE65 46968168 IC50 = 248 nM T13260 CKJ9S6 46968847 IC50 = 3100 nM T13260 CO2XL1 46970377 IC50 = 9 nM T13260 C0GZ4Q 46980515 IC50 = 498 nM T13260 C8QCH2 49779539 IC50 = 2.1 nM T13260 C7V2XL 49779540 IC50 = 0.25 nM T13260 CIC9S5 49799473 IC50 = 5750 nM T13260 C5ZNK0 49799653 IC50 = 21860 nM T13260 CZG04F 49799654 IC50 = 8490 nM T13260 CX5LZ9 50915159 IC50 = 0.018 nM T13260 C8N5OK 50991893 IC50 = 0.21 nM T13260 C0RUX1 50994677 IC50 > 10000 nM T13260 CL2O0Y 50994839 IC50 > 16200 nM T13260 CTG6R4 51041013 IC50 = 4400 nM T13260 CGX85M 51042201 IC50 = 30700 nM T13260 CWG69M 51042401 IC50 = 32300 nM T13260 C1AT4L 51042402 IC50 = 26800 nM T13260 C1VF4Z 51346982 IC50 = 0.015 nM T13260 C6Y3EL 51346989 IC50 = 0.015 nM T13260 C8GQS7 51351108 IC50 > 50000 nM T13260 CB8ND9 51354813 IC50 > 16900 nM T13260 CMXR96 51355428 IC50 = 114 nM T13260 C5KTL3 51355429 IC50 = 113 nM T13260 C4UTM8 51355430 IC50 = 130 nM T13260 CH5C9K 51355431 IC50 = 235 nM T13260 CRK2Q9 51355432 IC50 = 207 nM T13260 CF7RG5 51355433 IC50 = 141 nM T13260 C8XHD9 51355434 IC50 = 267 nM T13260 C41SUK 51355703 IC50 = 178 nM T13260 CM6T7H 51355704 IC50 = 127 nM T13260 CZDA87 51355705 IC50 = 481 nM T13260 CO1V0Y 51355706 IC50 = 169 nM T13260 C2OCG3 51355707 IC50 = 165 nM T13260 CGLU79 51355708 IC50 = 72 nM T13260 CL6XD4 51355709 IC50 = 72 nM T13260 C57MWS 51355970 IC50 = 292 nM T13260 CYC86A 51355971 IC50 = 690 nM T13260 CP7V3Q 51355972 IC50 = 112 nM T13260 CR6NH8 51355973 IC50 = 164 nM T13260 C6SD4P 51355974 IC50 = 296 nM T13260 C97MZT 51355975 IC50 = 81 nM T13260 CJU1O7 51355976 IC50 = 70 nM T13260 CIR0L7 51356252 IC50 = 47 nM T13260 C0BW7G 51356253 IC50 = 105 nM T13260 C39RVA 51356254 IC50 = 3750 nM T13260 C3P5LI 51356255 IC50 = 455 nM T13260 CKXR01 51356256 IC50 = 67 nM T13260 CF21EH 51356258 IC50 = 317 nM T13260 C4M5ZT 51356554 IC50 = 532 nM T13260 CS7X3R 51356555 IC50 = 4010 nM T13260 CR7UG9 51356556 IC50 = 313 nM T13260 C87FEB 51520434 IC50 = 600 nM T13260 C42JIQ 52912619 IC50 = 5040 nM T13260 CY0TF7 53237486 IC50 = 510 nM T13260 C5WQX4 53237725 IC50 = 1000 nM T13260 CD7HC1 53305315 IC50 = 91 nM T13260 C5SN8I 53317948 IC50 = 11000 nM T13260 CQZV41 53318733 IC50 = 30000 nM T13260 C9OPT6 53320278 IC50 = 0.75 nM T13260 CDM50Q 53320823 IC50 = 660 nM T13260 CRLJ68 53321508 IC50 = 700 nM T13260 CCNP36 53321604 IC50 = 0.47 nM T13260 CDV3X5 53323228 IC50 = 3600 nM T13260 C4WY6N 53323229 IC50 = 1000 nM T13260 CFC42O 53323677 IC50 > 16800 nM T13260 CFMK70 53324579 IC50 = 280 nM T13260 C48XBG 53325332 IC50 = 860 nM T13260 CA32FG 53325544 IC50 = 0.05 nM T13260 CN0SW9 53326827 IC50 = 0.1 nM T13260 CSQ45A 53326828 IC50 = 0.15 nM T13260 C0AL2O 53482563 IC50 = 11.8 nM T13260 C0P3VM 53637746 Ki = 58 nM T13260 CAE25J 53763992 IC50 = 970 nM T13260 CUXV34 54026593 Ki = 120 nM T13260 C53FSN 54165563 Ki = 7 nM T13260 C8FA6I 54348149 Ki = 58 nM T13260 CA19BF 54513089 Ki = 25 nM T13260 CE0PC5 54576531 IC50 = 4640 nM T13260 CS0NM1 54576532 IC50 = 1360 nM T13260 CA3YL8 54580402 IC50 = 5790 nM T13260 CB5QY9 54583302 IC50 = 34 nM T13260 CB02LJ 54584262 IC50 = 32 nM T13260 C34FYG 54584352 IC50 = 66.5 nM T13260 CLPG92 54586184 IC50 = 36 nM T13260 C91LBU 54597383 IC50 = 3300 nM T13260 C6G8HK 54597384 IC50 = 1800 nM T13260 CV2NS6 54729584 IC50 = 220 nM T13260 C70EIF 54756790 IC50 > 50000 nM T13260 CZU5L8 54768666 IC50 = 17340 nM T13260 C4C1ZY 54768667 IC50 = 10700 nM T13260 C5AVO9 54770656 IC50 = 12200 nM T13260 C2RW0G 54770885 IC50 = 12010 nM T13260 CW6EK4 54770886 IC50 = 4700 nM T13260 CTP0G9 54770887 IC50 = 5070 nM T13260 CHY71M 54770888 IC50 = 10600 nM T13260 CS42BX 54770889 IC50 = 16020 nM T13260 CU07HL 54770890 IC50 = 19320 nM T13260 CD2JA7 54770891 IC50 = 10330 nM T13260 CD1V8X 54771121 IC50 = 79980 nM T13260 CMX14D 54771122 IC50 = 10970 nM T13260 CVED14 54771123 IC50 = 16110 nM T13260 CPJW41 54771124 IC50 = 7730 nM T13260 C8JEH4 54771125 IC50 = 10950 nM T13260 CA4JF1 54771126 IC50 = 12160 nM T13260 C6Y8ND 54771341 IC50 = 10960 nM T13260 C7E3KS 54771342 IC50 = 14830 nM T13260 C6NRM1 54771343 IC50 = 19360 nM T13260 C3MR9N 54771344 IC50 = 13540 nM T13260 CI5QD9 54771345 IC50 = 13720 nM T13260 C7KBU3 54771346 IC50 = 12940 nM T13260 C7LOA4 54771347 IC50 = 31260 nM T13260 C8OI5N 54771563 IC50 = 13350 nM T13260 CUF4O0 54771564 IC50 = 13370 nM T13260 CP1UM5 54771565 IC50 = 16410 nM T13260 C3ZKB4 54771566 IC50 = 11610 nM T13260 C3YD8A 54771567 IC50 = 26770 nM T13260 C3URW8 54771568 IC50 = 15210 nM T13260 C2BYD3 54771787 IC50 = 4370 nM T13260 CUY87L 54771788 IC50 = 5260 nM T13260 C3WVO7 54771789 IC50 = 3070 nM T13260 CYM98K 54771790 IC50 = 7880 nM T13260 CV5S9D 54771791 IC50 = 10700 nM T13260 C2G6DW 54771792 IC50 = 6090 nM T13260 CHOT94 54771793 IC50 = 3910 nM T13260 CA49SQ 54771794 IC50 = 9160 nM T13260 CN2ES5 54772014 IC50 = 15480 nM T13260 C38PQF 54772015 IC50 = 5620 nM T13260 C3Q9YI 54772016 IC50 = 4170 nM T13260 C76QVG 54772017 IC50 = 2340 nM T13260 C5KI4U 54772018 IC50 = 11570 nM T13260 CR1YL2 54772019 IC50 = 7470 nM T13260 C1OQ4B 54772020 IC50 = 9530 nM T13260 CL7XJ4 54772021 IC50 = 7980 nM T13260 C06PFH 56598207 IC50 = 10500 nM T13260 CL4KT8 56610874 Ki = 8.2 nM T13260 C78MXU 56612673 Ki = 8.2 nM T13260 CV1ZO2 56632357 Ki = 90 nM T13260 C4N0WL 56645363 IC50 = 1021 nM T13260 C57NSZ 56645568 IC50 = 1268 nM T13260 C6PUX9 56645570 IC50 = 4513 nM T13260 CM94ZH 56664989 IC50 = 2780 nM T13260 CMU51H 56681975 IC50 = 2270 nM T13260 C7G5IR 56835177 Ki = 790 nM T13260 C5US1Z 56835178 Ki = 60 nM T13260 C3IZU1 56835179 Ki = 50 nM T13260 CRGX16 56837844 IC50 > 50000 nM T13260 C7M1OX 56837845 IC50 > 50000 nM T13260 CHCM56 56837846 IC50 > 50000 nM T13260 CX19AT 57327815 IC50 = 93 nM T13260 C0I2DY 57327816 IC50 = 59 nM T13260 CY58ZD 57330086 IC50 > 5000 nM T13260 C1C0FZ 57384102 Ki = 0.06 nM T13260 CLJ8A1 57384103 Ki = 0.65 nM T13260 C6I3AN 57390179 IC50 > 50000 nM T13260 C1ZB3N 57390180 IC50 > 50000 nM T13260 CH19RM 57390181 IC50 > 50000 nM T13260 CG2J7F 57390275 IC50 = 64500 nM T13260 C0VRP8 57391308 Ki = 12560 nM T13260 C3BKO8 57391309 Ki = 1482 nM T13260 CW3P7T 57391581 Ki = 100 nM T13260 CI1R4S 57391583 Ki = 250 nM T13260 CB02XQ 57391954 IC50 > 50000 nM T13260 C94BSM 57392056 IC50 = 63200 nM T13260 CJA4L1 57393085 Ki = 1722 nM T13260 CS6V8A 57393681 IC50 > 50000 nM T13260 CPN7Q2 57393682 IC50 > 50000 nM T13260 CV4S6C 57393683 IC50 > 50000 nM T13260 CR5I9O 57393684 IC50 > 50000 nM T13260 C5VDL7 57395400 IC50 > 50000 nM T13260 CC53MX 57395527 IC50 = 47300 nM T13260 CV08LN 57395659 IC50 = 986 nM T13260 CI6Q5O 57395660 IC50 = 304 nM T13260 CQ06KW 57395661 IC50 = 229 nM T13260 C48VIY 57396573 Ki = 5321 nM T13260 C2NML8 57396574 Ki = 8.2 nM T13260 C83ZIP 57396575 Ki = 82.54 nM T13260 C2F1TI 57397238 IC50 > 50000 nM T13260 C4O5DT 57397345 IC50 = 68100 nM T13260 CBL9Z1 57397346 IC50 = 58600 nM T13260 CXP68J 57397347 IC50 = 72000 nM T13260 C5VLB1 57398353 Ki = 35.12 nM T13260 C4DE6B 57398582 Ki = 1000 nM T13260 CW2J6Z 57398927 IC50 > 50000 nM T13260 CP65RI 57398928 IC50 > 50000 nM T13260 CHB0A3 57398929 IC50 > 50000 nM T13260 C81RCO 57398930 IC50 > 50000 nM T13260 CD4BN7 57400011 Ki = 285.1 nM T13260 CJT2G9 57400012 Ki = 100 nM T13260 CJZX60 57400626 IC50 > 50000 nM T13260 CV8KD9 57400627 IC50 > 50000 nM T13260 C3G4RJ 57400766 IC50 = 44800 nM T13260 C2WJ7Y 57400842 IC50 = 57400 nM T13260 C5OYK8 57400879 IC50 = 114 nM T13260 CHVG47 57401821 Ki = 15000 nM T13260 C1MF0V 57402418 IC50 > 50000 nM T13260 CQ9C3L 57402419 IC50 = 26500 nM T13260 CUD85V 57402656 IC50 = 523 nM T13260 CD2U9L 57403526 Ki = 1160 nM T13260 CFI0L8 57403527 Ki = 3.17 nM T13260 C10SAL 57403795 Ki = 79.43 nM T13260 CRL10W 57413872 Ki = 86 nM T13260 C04MZQ 57520593 IC50 = 17000 nM T13260 CX8Q7H 57520594 IC50 = 5800 nM T13260 CYHS09 57679076 IC50 >= 200000 nM T13260 C7OK1X 57775654 IC50 = 4490 nM T13260 CQ0M7J 58215635 IC50 = 3400 nM T13260 C34JIZ 58255359 IC50 = 2130 nM T13260 C2TUJ7 58255382 IC50 = 228 nM T13260 C3DPC0 58255407 IC50 = 43 nM T13260 C9DK1X 58255415 IC50 = 488 nM T13260 CTI0D7 58255435 IC50 = 880 nM T13260 CRQ70M 58255438 IC50 > 500 nM T13260 CLQ65O 58255479 IC50 > 5000 nM T13260 CP6RA9 58255482 IC50 = 3073 nM T13260 CJX70M 58255566 IC50 = 105 nM T13260 CW71EO 58255581 IC50 = 447 nM T13260 C6XPA7 59356082 IC50 = 24000 nM T13260 CX2US1 59356084 IC50 = 35000 nM T13260 CD31PM 59356085 IC50 = 99000 nM T13260 CVRT12 59356087 IC50 = 41000 nM T13260 CLP2O3 60151424 IC50 = 6200 nM T13260 C9M4QI 60156307 IC50 = 112.3 nM T13260 CZ1WU8 60166590 IC50 = 169.3 nM T13260 CB7N8A 60195126 IC50 = 17 nM T13260 CE18JH 60202715 Ki = 48 nM T13260 CX4N0I 62707515 IC50 = 48 nM T13260 C0G3LA 66559847 IC50 = 49 nM T13260 C4RSI6 66559935 IC50 = 162 nM T13260 CDX7I8 66559936 IC50 = 22 nM T13260 CF9EQ5 66559939 IC50 = 2901 nM T13260 CQN6D3 66559940 IC50 = 394 nM T13260 CN4H8G 66559941 IC50 = 954 nM T13260 CTP6Q4 66559942 IC50 = 275 nM T13260 C9EGW2 66575742 IC50 > 10000 nM T13260 CMXA10 66575743 IC50 > 10000 nM T13260 CKWB91 66575744 IC50 > 10000 nM T13260 C7I3MW 66575745 IC50 > 10000 nM T13260 CPN17S 66575746 IC50 > 10000 nM T13260 CG0ZA7 66575747 IC50 > 10000 nM T13260 C6HF0U 66575748 IC50 > 10000 nM T13260 CDI93T 66575817 IC50 > 10000 nM T13260 CBP6I7 66576773 IC50 > 10000 nM T13260 C4NYB0 66576930 IC50 > 10000 nM T13260 C3LP5H 66576931 IC50 > 10000 nM T13260 CE03WG 66576932 IC50 > 10000 nM T13260 C9XYA1 67205290 Ki = 700 nM T13260 CO8IZ3 67854245 IC50 = 590 nM T13260 C2F5TS 68037237 Ki = 442 nM T13260 C97FZU 68561433 IC50 = 31 nM T13260 CK05PZ 68668617 Ki = 7 nM T13260 CC75HS 69198620 IC50 = 160000 nM T13260 CI6U5W 69649421 IC50 = 160 nM T13260 CZN04V 69828765 Ki = 45 nM T13260 CSUX85 70178310 Ki = 55 nM T13260 CBM80I 70354859 Ki = 77 nM T13260 COGQ93 70680979 IC50 = 30000 nM T13260 C96QKR 70683101 IC50 = 61000 nM T13260 CBNF56 70689398 IC50 = 20000 nM T13260 CPNR72 70689399 IC50 = 32000 nM T13260 CCG0U6 70691503 IC50 = 18000 nM T13260 CKE71B 70691504 IC50 = 11000 nM T13260 CA36IC 70695715 IC50 = 29000 nM T13260 CHEJ23 70748349 IC50 = 20900 nM T13260 C1VMF2 70977969 IC50 > 10000 nM T13260 CUV23H 71449132 Ki = 22 nM T13260 C37CSD 71450101 IC50 = 181.1 nM T13260 C7EDZ9 71452741 Ki = 753 nM T13260 CFKO73 71453732 IC50 = 2180 nM T13260 CI6B9U 71454429 IC50 > 50000 nM T13260 C70TUP 71455138 IC50 = 11 nM T13260 CH70RK 71456229 IC50 = 11000 nM T13260 CFG4L5 71456934 IC50 = 35 nM T13260 C8NPL7 71457257 IC50 = 83 nM T13260 CJCY84 71457258 IC50 = 20 nM T13260 C1KY3Q 71458062 Ki = 86 nM T13260 CK5TV7 71461661 Ki = 206 nM T13260 CI16NC 71520311 IC50 = 32 nM T13260 CE9A6B 71520312 IC50 = 246 nM T13260 C03VKJ 71520313 IC50 > 5000 nM T13260 C5J7DI 71520314 IC50 = 3340 nM T13260 CE0N5C 71520315 IC50 > 5000 nM T13260 C4Z6YP 71520316 IC50 = 565 nM T13260 CC8Z6L 71520431 IC50 > 5000 nM T13260 C1DK9P 71520432 IC50 = 1500 nM T13260 C9NOQ1 71521632 IC50 = 2130 nM T13260 C0OTA2 71521716 IC50 = 3660 nM T13260 CVLE07 71521717 IC50 > 5000 nM T13260 CJKX84 71521718 IC50 = 1350 nM T13260 CZ5P9U 71521719 IC50 = 140 nM T13260 C1YCB0 71521720 IC50 = 889 nM T13260 CE57PM 71521721 IC50 = 74 nM T13260 C0O2SA 71521798 IC50 = 81 nM T13260 CMEC10 71521799 IC50 = 59 nM T13260 CR9O5T 71521800 IC50 = 273 nM T13260 C0JBI3 71521801 IC50 = 74 nM T13260 CE7Z4I 71521802 IC50 = 116 nM T13260 CW2AG4 71521803 IC50 = 19 nM T13260 C6ID7K 71521804 IC50 = 55 nM T13260 CPZ5S8 71535400 IC50 = 790 nM T13260 CCRS95 71535683 IC50 = 2200 nM T13260 C9V7KW 71568307 IC50 = 9.01 nM T13260 CZGA56 71568308 IC50 = 148.93 nM T13260 C0E3WP 71568309 IC50 = 77.36 nM T13260 C3IX0R 71568310 IC50 = 4.93 nM T13260 C1B6UY 71568311 IC50 = 16.58 nM T13260 CF6DO2 71568312 IC50 = 21.39 nM T13260 CNBX98 71568313 IC50 = 164.01 nM T13260 CLD9N8 71568314 IC50 = 138.72 nM T13260 C7YVC9 71568442 IC50 = 56.83 nM T13260 C2ZS4G 71568443 IC50 = 27.01 nM T13260 C2BD6R 71568444 IC50 = 6.23 nM T13260 C03WJE 71568445 IC50 = 48.93 nM T13260 CXH93O 71568446 IC50 = 25.56 nM T13260 C0N6UG 71568447 IC50 = 46.92 nM T13260 C3PZG5 71568448 IC50 = 57.43 nM T13260 CPI06S 71568584 IC50 = 111.09 nM T13260 CL4YR2 71568585 IC50 = 203.34 nM T13260 C7ZCL4 71568586 IC50 = 235.33 nM T13260 CTQ79Z 71568587 IC50 = 217.43 nM T13260 C58SMB 71574941 IC50 = 480 nM T13260 CC09FQ 71574942 IC50 = 460 nM T13260 CA2T5L 71574943 IC50 = 300 nM T13260 C9MFZ7 71574944 IC50 = 1100 nM T13260 CW73OE 71574945 IC50 = 1973 nM T13260 C70NHJ 71574946 IC50 = 400 nM T13260 CLH83S 71574947 IC50 = 837 nM T13260 CF71AB 71575030 IC50 = 575 nM T13260 CCG1S5 71575031 IC50 = 565 nM T13260 CH9WE7 71575032 IC50 = 260 nM T13260 CO4ZQ7 71575033 IC50 = 170 nM T13260 CT86GV 71575034 IC50 = 6393 nM T13260 CHC8L4 71614085 IC50 = 0.2 nM T13260 CKPV51 71621803 IC50 > 100000 nM T13260 CG72JK 71681355 IC50 = 9257 nM T13260 C56LUJ 71716957 IC50 = 11160 nM T13260 CJE01S 71745100 IC50 > 10000 nM T13260 C54KVE 71748876 IC50 = 670 nM T13260 CT5Q9N 71812321 IC50 = 750 nM T13260 CBL42N 71812322 IC50 = 450 nM T13260 C9IOA1 71812324 Ki = 45 nM T13260 CX0WV5 71817943 IC50 > 2000 nM T13260 CN1LU6 71817944 IC50 > 2000 nM T13260 CGV4U3 71817945 IC50 > 2000 nM T13260 CJ4L5G 71818086 IC50 > 2000 nM T13260 COXA51 71818087 IC50 > 2000 nM T13260 CP1A3M 71818088 IC50 > 2000 nM T13260 CPJ42T 71818089 IC50 > 2000 nM T13260 CAP03I 71818090 IC50 > 2000 nM T13260 CO23PK 71818091 IC50 > 2000 nM T13260 CL4X6A 71818092 IC50 > 2000 nM T13260 CL8GK5 71818093 IC50 > 2000 nM T13260 C4ZVG0 71818094 IC50 > 2000 nM T13260 CH2GR0 71818232 IC50 > 2000 nM T13260 C0VGQ9 71818233 IC50 > 2000 nM T13260 C5QRF2 71818234 IC50 > 2000 nM T13260 C09VHD 72194216 IC50 = 5500 nM T13260 C4POE7 72546693 Ki = 80 nM T13260 CKI39Q 72546694 Ki = 20 nM T13260 C2SE6Q 72546935 Ki = 111 nM T13260 C49MBW 72546936 Ki = 160 nM T13260 CJCU54 72546937 Ki = 70 nM T13260 CN1Z5U 72546938 Ki = 20 nM T13260 CD6I2S 72546939 Ki = 330 nM T13260 CKE4O3 72546940 Ki = 170 nM T13260 CW5H8C 72546941 Ki = 820 nM T13260 C74PHD 72547200 Ki = 200 nM T13260 CDC4P8 72547201 Ki = 130 nM T13260 CZNW37 72547202 Ki = 841 nM T13260 CFLU42 72547203 Ki = 110 nM T13260 C76AZT 72547204 Ki = 90 nM T13260 C1IP7G 72547205 Ki = 237 nM T13260 C62CNP 72547206 Ki = 350 nM T13260 CG0LT8 72547452 Ki = 647 nM T13260 CU76NM 72703468 IC50 > 10000 nM T13260 C9PRT7 72703681 IC50 > 10000 nM T13260 CCG7R3 72703685 IC50 = 5.3 nM T13260 CU27CK 72703887 IC50 > 10000 nM T13260 CFR2V8 72703888 IC50 > 10000 nM T13260 CAU4Z0 72703889 IC50 = 3.1 nM T13260 C56KEC 72703890 IC50 = 13.3 nM T13260 CB7PR0 72704087 IC50 = 1472 nM T13260 C5SNU6 72708597 IC50 = 3200 nM T13260 CSB7R2 73055580 IC50 = 15000 nM T13260 CG37VI 73055876 IC50 = 20000 nM T13260 CU5DC1 73055877 IC50 = 190000 nM T13260 C5M7RH 73055879 IC50 = 2500 nM T13260 C53JKM 73055880 IC50 = 67100 nM T13260 CR8V7S 73055881 IC50 = 800 nM T13260 C72LFY 73346265 IC50 = 2700 nM T13260 C5F2VZ 73347760 IC50 = 3400 nM T13260 C5QTA7 73349312 IC50 = 3400 nM T13260 CPU7N5 73350879 IC50 = 12500 nM T13260 CT1J5B 73350882 IC50 = 12500 nM T13260 C9Y5FN 73353441 IC50 = 9257 nM T13260 CT9SN8 73353827 IC50 = 4600 nM T13260 CD13BV 73353828 IC50 = 8000 nM T13260 CGWY15 73355361 IC50 = 1800 nM T13260 C1YT7X 73355362 IC50 = 9400 nM T13260 CKEY08 73355363 IC50 = 7900 nM T13260 CGF87Z 73355403 IC50 = 3900 nM T13260 C0OY5P 73356914 IC50 = 1300 nM T13260 CX12ML 73356915 IC50 = 2900 nM T13260 C0UQ3M 73356955 IC50 = 29100 nM T13260 CKG8J2 73357190 IC50 = 590 nM T13260 C9WY3B 73386689 IC50 = 45 nM T13260 CK4NQ1 76186646 IC50 = 0.9 nM T13260 CM52SI 76308995 IC50 = 11900 nM T13260 CS80JY 76310075 IC50 = 50 nM T13260 CB1V2S 76311295 IC50 = 10700 nM T13260 C7XH3E 76314886 IC50 = 80 nM T13260 CPU3T6 76317295 IC50 = 1100 nM T13260 CAM49B 76318503 IC50 = 90 nM T13260 CFJ8G5 76322165 IC50 = 40 nM T13260 C7KEG3 76322166 IC50 = 150 nM T13260 CHBR20 76325787 IC50 = 1010 nM T13260 CXD53T 76327865 IC50 = 160 nM T13260 CS8D4U 76328231 IC50 = 3000 nM T13260 C3F0JZ 76329384 IC50 > 300000 nM T13260 C3JID2 76331906 IC50 = 650 nM T13260 C1YJW0 77846787 IC50 = 790 nM T13260 CV73PD 77846790 IC50 = 10000 nM T13260 C0DIH7 77846872 IC50 = 10000 nM T13260 COI25M 77846873 IC50 = 1000 nM T13260 CJI8R0 77846875 IC50 = 3800 nM T13260 CZK4J1 77846962 IC50 = 2800 nM T13260 CEK89G 77846963 IC50 = 10000 nM T13260 C5BA8Z 77846964 IC50 = 1240 nM T13260 C4D6XJ 77847803 IC50 = 1600 nM T13260 CF7O4Q 77847804 IC50 = 1200 nM T13260 CEC49D 85863219 IC50 = 1610 nM T13260 CZ5PM0 86277538 IC50 = 0.42 nM T13260 CHV8R6 86307678 IC50 = 620 nM T13260 C3X6MJ 86792466 IC50 = 21700 nM T13260 CL30TR 89471870 IC50 = 2300 nM T13260 C3BUS8 89471889 IC50 = 420 nM T13260 CI7HY8 89471890 IC50 = 120 nM T13260 CX0M7B 89961716 IC50 = 21 nM T13260 CR5D6Y 89961785 IC50 > 10000 nM T13260 C89TEU 89968659 IC50 > 10000 nM T13260 CY5IC7 90252834 IC50 = 4600 nM T13260 C84NVA 90252850 IC50 = 6300 nM T13260 CBY46O 90252851 IC50 = 5400 nM T13260 CNVA50 90252852 IC50 = 6200 nM T13260 C89BFG 90333640 IC50 = 1820 nM T13260 CJ8NI5 90655716 Ki = 57 nM T13260 COF02L 90655717 Ki = 62 nM T13260 CO9K2W 90655718 Ki = 31 nM T13260 CX8L7D 90655719 Ki = 69 nM T13260 CHD21I 90666137 IC50 = 14.4 nM T13260 C4A7JU 90677206 IC50 = 12500 nM T13260 C3T5BI 90677209 IC50 = 12500 nM T13260 CV96EW 90677213 IC50 = 12500 nM T13260 C3Y8AQ 90677215 IC50 = 12500 nM T13260 C6PJL5 90677216 IC50 = 12500 nM T13260 CFI3J8 90677218 IC50 = 12500 nM T13260 CQ91ZO 90677219 IC50 = 12500 nM T13260 CQS8C9 91664365 IC50 = 1000 nM T13260 CM9U7B 91758284 Ki = 20 nM T13260 CLB2E7 91827654 IC50 > 30000 nM T13260 C0KDB6 91983064 Ki = 32 nM T13260 CYL1S3 97191385 IC50 = 5100 nM T13260 CXRB41 101152219 IC50 > 10000 nM T13260 C3P9ZY 101199629 IC50 = 41 nM T13260 CL3UQ9 101354484 Ki = 10 nM T13260 C26AKT 101354485 Ki = 14 nM T13260 CZXS85 101354486 Ki = 81 nM T13260 CWXT16 101378163 Ki = 45 nM T13260 C8VZC7 101378164 Ki = 45 nM T13260 C4G5MB 101378165 Ki = 670 nM T13260 C5HLB7 101378166 Ki = 670 nM T13260 C0TOW6 101433013 Ki = 8.2 nM T13260 CLI59T 101579737 IC50 = 160 nM T13260 C18UTF 101587707 Ki = 150 nM T13260 C2SUC3 101587708 Ki = 1180 nM T13260 CI0N8C 101592374 Ki = 24.1 nM T13260 CV87DF 101592375 Ki = 24.1 nM T13260 C1ZN6O 101592376 Ki = 24.1 nM T13260 C5WGQ7 101620856 Ki = 5000 nM T13260 CC01NA 101650066 Ki = 12 nM T13260 CE9T0K 101650068 Ki = 12 nM T13260 CUDV46 101650069 Ki = 12 nM T13260 CBN09G 101651130 Ki = 2 nM T13260 C9CZN6 101668720 Ki = 11100 nM T13260 C9TID7 101701780 Ki = 5000 nM T13260 C0RN1M 101927481 Ki = 25 nM T13260 C9E7GV 102068512 Ki = 7 nM T13260 C63RAU 102068514 Ki = 7 nM T13260 C8YJK2 102068516 Ki = 7 nM T13260 C57AZV 102068518 Ki = 7 nM T13260 C4J1SX 102279741 Ki = 95 nM T13260 CE90MX 102346108 IC50 = 6870 nM T13260 CED87Z 102439715 Ki = 5000 nM T13260 C0DYC5 102532604 Ki = 5000 nM T13260 C9KZ5G 102533756 Ki = 16 nM T13260 CB1Z8U 102533759 Ki = 16 nM T13260 CMO84S 110730849 IC50 = 490 nM T13260 CJ9Z0S 118496546 IC50 = 6900 nM T13260 C2BMT8 118708021 IC50 = 34400 nM T13260 C8NES2 118711691 Ki = 630.96 nM T13260 CKT4A8 118711692 Ki = 707.95 nM T13260 COD91Y 118711693 Ki = 707.95 nM T13260 CGJ93V 118711694 Ki = 25.12 nM T13260 C0WLI2 118711695 Ki = 354.81 nM T13260 CXDE52 118711696 Ki = 144.54 nM T13260 CAW5K3 118723935 IC50 = 549 nM T13260 CK8UL1 118723936 IC50 = 387 nM T13260 CIW7O0 118723937 IC50 = 477 nM T13260 C42CEZ 118723938 IC50 = 584 nM T13260 CJQ63E 118723939 IC50 = 639 nM T13260 CCXN71 118723940 IC50 = 445 nM T13260 CS78BD 118723941 IC50 = 349 nM T13260 C9W3QX 118723942 IC50 = 17464 nM T13260 COJ2K8 118723943 IC50 = 5855 nM T13260 CZ23UL 118723944 IC50 = 3708 nM T13260 CIWU64 118723945 IC50 = 4566 nM T13260 CZI6A0 118723946 IC50 = 8299 nM T13260 COB46M 118723947 IC50 = 31813 nM T13260 CJ1HP9 118728223 Ki = 10000 nM T13260 CZR62N 118730170 IC50 = 810 nM T13260 CDHI10 118733086 IC50 > 10000 nM T13260 C18PWB 118733087 IC50 > 10000 nM T13260 C8WJ2Y 118733088 IC50 > 10000 nM T13260 C31ZXP 118733089 IC50 > 10000 nM T13260 CHR84E 118733090 IC50 > 10000 nM T13260 CAQ72M 118733091 IC50 > 10000 nM T13260 CIV1Z5 118733092 IC50 > 10000 nM T13260 CU3Y9W 118733093 IC50 > 10000 nM T13260 CF49NU 118733094 IC50 > 10000 nM T13260 CK73VU 118733095 IC50 > 10000 nM T13260 CR1WU5 118733096 IC50 > 10000 nM T13260 C5C4FZ 118735165 IC50 = 447 nM T13260 C1ZLM6 118735166 IC50 = 146 nM T13260 CQXM57 118735167 IC50 = 75 nM T13260 C0RYM4 118735168 IC50 = 137 nM T13260 C0DCB9 118735169 IC50 = 2425 nM T13260 CG4QF3 118735170 IC50 = 1894 nM T13260 CD3IY5 118735171 IC50 = 4993 nM T13260 C2VJU4 118735179 IC50 = 2090 nM T13260 CXWH51 118735180 IC50 = 165 nM T13260 C3YUS9 118735181 IC50 = 1546 nM T13260 CZET62 118735186 IC50 = 128 nM T13260 CZ8U2C 118735187 IC50 = 157 nM T13260 COJ81W 118735362 IC50 = 1020 nM T13260 C8VFT2 118735363 IC50 = 1320 nM T13260 CZE92I 118735364 IC50 = 53.1 nM T13260 CFB1G7 118735365 IC50 = 48.1 nM T13260 CX4V1E 118735366 IC50 = 6290 nM T13260 CW60ZD 118735367 IC50 = 337 nM T13260 C6ULM1 118735368 IC50 = 143 nM T13260 CE50LC 118735369 IC50 = 261 nM T13260 CMCW85 118735370 IC50 = 328 nM T13260 C6Y2NQ 118735371 IC50 = 1930 nM T13260 CVEQ39 118735372 IC50 = 48.9 nM T13260 C4LK0C 118735373 IC50 = 16.9 nM T13260 C93CNO 118735374 IC50 = 174 nM T13260 C4YR6E 118735375 IC50 = 715 nM T13260 CS3ZJ8 118735376 IC50 = 699 nM T13260 CV83KA 118735377 IC50 = 493 nM T13260 C0BP6M 118735378 IC50 = 30500 nM T13260 CG9RB4 118735379 IC50 = 1240 nM T13260 CGT60X 118735380 IC50 = 7340 nM T13260 CY6L8W 118735381 IC50 = 491 nM T13260 C3NB6I 122181247 IC50 = 12500 nM T13260 CYCG69 122181248 IC50 = 200 nM T13260 CME27L 122181249 IC50 = 1800 nM T13260 C0KHC3 122191579 IC50 = 0.26 nM T13260 CO7E3N 122191580 IC50 = 0.42 nM T13260 CML6C5 122191581 IC50 = 5.2 nM T13260 CYC63O 122191582 IC50 = 2.7 nM T13260 CP7S0B 122191583 IC50 = 2.3 nM T13260 C61IRT 122191584 IC50 = 4 nM T13260 CYJ32S 122191585 IC50 = 2.3 nM T13260 CAQ5S2 122191586 IC50 = 3.5 nM T13260 C03SBU 122191587 IC50 = 4.2 nM T13260 CLG6J4 122191588 IC50 = 5 nM T13260 CI42KY 122191589 IC50 = 20.7 nM T13260 C9GQP6 122191591 IC50 = 3.4 nM T13260 C0WN2U 122191592 IC50 = 5.5 nM T13260 C0WI6K 122191772 IC50 = 29 nM T13260 C5C2EM 122192355 IC50 = 250 nM T13260 C4HIF8 122192356 IC50 = 220 nM T13260 C0SJU6 122192359 IC50 = 100 nM T13260 C3T9CZ 122192360 IC50 = 41 nM T13260 C58OCL 122192361 IC50 = 0.1 nM T13260 C15NCI 122439267 IC50 = 10000 nM T13260 CX4T7L 122439274 IC50 = 10000 nM T13260 C3YG1J 122443028 IC50 > 19952.62 nM T13260 CW3K8X 122462796 IC50 > 19952.62 nM T13260 C80OLS 122462854 IC50 > 31622.78 nM T13260 CR4YC2 124012328 Ki = 38 nM T13260 C10TQU 124351848 Ki = 1 nM T13260 CCX94N 124351849 Ki = 75 nM T13260 C36AXJ 127025738 Ki = 100 nM T13260 CM2NC0 127025739 Ki = 100 nM T13260 CW5AZ0 127025740 Ki = 100 nM T13260 CY9Q8T 127025741 Ki = 100 nM T13260 C0X8HP 127026020 Ki = 24.1 nM T13260 C4LWG3 127026653 IC50 = 120500 nM T13260 C3ZQ5Y 127026654 IC50 = 1889 nM T13260 CZDU19 127026655 IC50 = 18570 nM T13260 CIT8S3 127026966 IC50 = 1820 nM T13260 CJTB10 127026967 IC50 = 1820 nM T13260 C2ZFR8 127027572 IC50 = 7900 nM T13260 CV1BD6 127027573 IC50 = 3100 nM T13260 C1L9TB 127027959 IC50 = 26000 nM T13260 CPX6K3 127028274 Ki = 100 nM T13260 CQO36B 127028499 IC50 = 5000 nM T13260 CCR07G 127028593 IC50 = 1820 nM T13260 CH6PU4 127028608 Ki = 100 nM T13260 C9WIB4 127028609 Ki = 100 nM T13260 CN42BR 127028817 IC50 > 10000 nM T13260 CIE4Q7 127028911 IC50 = 1820 nM T13260 C49IME 127031799 IC50 = 6100 nM T13260 CGEO60 127035149 IC50 = 245 nM T13260 CJ30BZ 127035150 IC50 = 236 nM T13260 C3MN9I 127035661 Ki = 5 nM T13260 CX3TB1 127035807 Ki = 5 nM T13260 CE6T8A 127035808 Ki = 5 nM T13260 C7JNM3 127036045 Ki = 75000 nM T13260 CS72ZI 127036174 Ki = 100 nM T13260 C9AFT8 127036253 IC50 = 6400 nM T13260 CQS2U0 127036843 IC50 = 2800 nM T13260 C7SM8Y 127037253 Ki = 31 nM T13260 CW08IP 127037254 IC50 = 1700 nM T13260 CXWJ74 127037557 Ki = 36 nM T13260 CK5N0X 127037559 Ki = 10000 nM T13260 CMQD16 127037560 Ki = 10000 nM T13260 CI6S7D 127037561 Ki = 10000 nM T13260 CTE51A 127047976 IC50 = 110 nM T13260 C1IBC5 127048009 IC50 = 530 nM T13260 CWE96C 127048149 IC50 = 12310 nM T13260 CDX0L1 127048499 IC50 = 51 nM T13260 CWD0J9 127048833 IC50 = 7 nM T13260 C9OEW2 127048838 IC50 = 46 nM T13260 CCJ3F0 127048839 IC50 = 6 nM T13260 CQ10PX 127048840 IC50 = 42 nM T13260 CWAH54 127048841 IC50 = 48 nM T13260 CD2O0K 127049168 IC50 = 129 nM T13260 C7ZHU6 127049169 IC50 = 48 nM T13260 CQN95D 127049828 IC50 = 36 nM T13260 C20LNJ 127050749 IC50 = 43 nM T13260 CH6E4C 127050950 IC50 = 168 nM T13260 CQ8PA9 127050951 IC50 = 512 nM T13260 C4Q6RA 127050952 IC50 = 800 nM T13260 C92CDW 127051351 IC50 = 14 nM T13260 CCR94D 127051352 IC50 = 13 nM T13260 CPL7A6 127051353 IC50 = 54 nM T13260 C7T2JR 127051680 IC50 = 339 nM T13260 CEJ1B8 127051681 IC50 = 131 nM T13260 CW3B0L 127051682 IC50 = 79 nM T13260 CE04JD 127052583 IC50 = 16 nM T13260 C48EUT 127052584 IC50 = 45 nM T13260 CT73HY 127052585 IC50 = 21 nM T13260 CL4ZK7 127052586 IC50 = 59 nM T13260 C1EI2R 127052880 IC50 = 22 nM T13260 CU9FI0 127052881 IC50 = 14 nM T13260 C01SHM 127052902 IC50 = 53 nM T13260 C09AZE 127052903 IC50 = 24 nM T13260 CH85FP 127052904 IC50 = 14 nM T13260 CYVM52 127052905 IC50 = 9 nM T13260 C12WOQ 129137247 IC50 = 62.2 nM T13260 C4O3QV 129137260 IC50 = 177.1 nM T13260 CJB4M3 129137266 IC50 = 230 nM T13260 CWVE96 129137276 IC50 = 13.4 nM T13260 CJ1N2M 129137280 IC50 = 220.8 nM T13260 CH42QX 129137285 IC50 = 8.8 nM T13260 CEH4N6 129750903 IC50 = 2600 nM T13260 CD7BX2 132601756 IC50 = 57.54 nM T13260 C5XSM4 132601757 IC50 = 12.11 nM T13260 CC2X1M 132601758 IC50 = 9.016 nM T13260 C8U1VZ 132601759 IC50 = 17.38 nM T13260 CH3V9Q 134139925 IC50 = 7700 nM T13260 CZV71F 134140768 IC50 = 6070 nM T13260 CVS3Q5 134142034 IC50 = 9724 nM T13260 CK4GS1 134142054 IC50 = 4660 nM T13260 C4B3MJ 134142750 IC50 = 9520 nM T13260 C2PT7N 134146686 IC50 = 12530 nM T13260 CK1BE9 134155077 IC50 = 286.9 nM T13260 C8QEA7 134155257 IC50 = 5089 nM T13260 C2BK3Z 134155779 IC50 = 645.3 nM T13260 C6G1CH 135185858 IC50 = 6445 nM T13260 CVR24H 135461648 IC50 = 29800 nM T13260 COWK61 135926058 IC50 > 50000 nM T13260 C7MP6W 135967555 Ki = 2548 nM T13260 CAV9U3 136219390 IC50 = 11.4 nM T13260 C59TUZ 136239410 IC50 > 10000 nM T13260 CH0O1B 136239411 IC50 > 10000 nM T13260 C52CVP 136239516 IC50 = 4152 nM T13260 CC7LY3 136239517 IC50 = 454 nM T13260 CSQR53 136239518 IC50 = 2112 nM T13260 C1N2WP 136244527 IC50 = 6195 nM T13260 C2V0IM 136244612 IC50 = 6 nM T13260 CLU5W1 136244613 IC50 = 922 nM T13260 C5LFY4 136245940 IC50 > 10000 nM T13260 CF07BL 136245941 IC50 > 10000 nM T13260 CYIF59 136245971 IC50 > 10000 nM T13260 CM6GS7 137632939 IC50 = 8900 nM T13260 CD7J1Z 137635610 IC50 = 5670 nM T13260 C4FYB7 137650013 IC50 = 9670 nM T13260 C2OC5D 137660208 IC50 = 6700 nM T13260 C3UK1Z 137660483 IC50 > 10000 nM T13260 C6VX2G 137662301 IC50 = 30.3 nM T13260 CEG7C9 140993853 IC50 = 1092.68 nM T13260 CY9QN0 145949171 IC50 = 2700 nM T13260 C0R6GF 145949298 IC50 = 237.6 nM T13260 C51BOX 145949540 IC50 = 700 nM T13260 C8T1HG 145949588 IC50 = 677.4 nM T13260 CBR4W8 145950208 IC50 = 2700 nM T13260 CVIW14 145950556 IC50 = 2800 nM T13260 C3L5IO 145950622 IC50 = 2300 nM T13260 C2EN9P 145950803 IC50 = 2500 nM T13260 CH80BF 145951156 IC50 = 32.3 nM T13260 CE8S3P 145951478 IC50 = 11900 nM T13260 CF2JT9 145951520 IC50 = 51.2 nM T13260 CD9G1O 145951806 IC50 = 2635 nM T13260 CL7V8M 145952266 IC50 = 11200 nM T13260 C9J0MP 145952426 IC50 = 1058 nM T13260 C4RX0H 145952545 IC50 = 276.8 nM T13260 CAD1R5 145953186 IC50 = 82.9 nM T13260 CGTW16 145953426 IC50 = 9800 nM T13260 C3PG4W 145953645 IC50 = 9800 nM T13260 CCF34U 145954042 IC50 = 8300 nM T13260 C8AR7H 145954077 IC50 = 5500 nM T13260 C5J7MO 145954302 IC50 = 4400 nM T13260 C6LU3T 145954433 IC50 = 7600 nM T13260 CRZ51Q 145954497 IC50 = 217.4 nM T13260 CEU5V2 145955100 IC50 = 4200 nM T13260 CGH62B 145955360 IC50 = 3900 nM T13260 CV49CR 145955375 IC50 = 11900 nM T13260 CYZ7R9 145955426 IC50 = 1400 nM T13260 C04FSJ 145955438 IC50 = 4600 nM T13260 CV5CZ7 145955551 IC50 = 207.5 nM T13260 CO3P9B 145955618 IC50 = 1300 nM T13260 CPS1E4 145956015 IC50 = 14.1 nM T13260 CCVP89 145956394 IC50 = 108.7 nM T13260 CR79QW 145956423 IC50 = 3400 nM T13260 CH8KZ4 145956588 IC50 = 260.8 nM T13260 CF4X3A 145956605 IC50 = 5400 nM T13260 CP65IV 145957520 IC50 = 8800 nM T13260 C7VQ6H 145958289 IC50 = 3500 nM T13260 CW8K2X 145958349 IC50 = 196.5 nM T13260 C8COZ7 145958369 IC50 = 4000 nM T13260 CC7UM6 145958531 IC50 = 36.1 nM T13260 C7TS3W 145958716 IC50 = 7772 nM T13260 C1FBC3 145958737 IC50 = 58.3 nM T13260 C0X5WO 145958928 IC50 = 96.9 nM T13260 C5IEV3 145958952 IC50 = 800 nM T13260 CTGM23 145959211 IC50 = 2300 nM T13260 CV1N0L 145959349 IC50 = 3800 nM T13260 C62HPO 145959622 IC50 = 2800 nM T13260 C4NYX7 145959688 IC50 = 210.6 nM T13260 CCW9R3 145959703 IC50 = 4100 nM T13260 C90VNG 145960023 IC50 = 3200 nM T13260 C7HA8N 145960331 IC50 = 3500 nM T13260 CK71RV 145963932 IC50 > 31622.78 nM T13260 C79FGQ 145965325 IC50 > 31622.78 nM T13260 CI56TJ 145967693 IC50 = 935.46 nM T13260 CKWV62 145967722 IC50 = 3591.14 nM T13260 C7XT0Z 145967929 IC50 = 3482.15 nM T13260 CHA9G8 145967940 IC50 = 3045.68 nM T13260 C0HP1U 145968036 IC50 = 2600.71 nM T13260 C5BM1L 145968186 IC50 = 999.74 nM T13260 C8XB7E 145968768 IC50 = 3253.28 nM T13260 C4JM2H 145968847 IC50 = 5715.79 nM T13260 C74IZW 145969198 IC50 = 3187.68 nM T13260 CNV0K1 145969871 IC50 = 1181.36 nM T13260 C4MQL6 145970012 IC50 = 1984.4 nM T13260 CDZV35 145970043 IC50 = 176.82 nM T13260 CEKI13 145970456 IC50 = 3321.79 nM T13260 C2Q1CO 145970604 IC50 = 1804.56 nM T13260 CW7XA4 145970723 IC50 = 3565.19 nM T13260 CE6P4U 145971254 IC50 = 1700 nM T13260 CGBW36 145972890 IC50 = 15300 nM T13260 CR50XP 145974563 IC50 = 54.4 nM T13260 CTB32X 145987737 IC50 = 3000.88 nM T13260 CJQ23A 145988166 IC50 = 3345.23 nM T13260 CAS5W8 145988425 IC50 = 3409.25 nM T13260 CZBY26 145988625 IC50 = 1703.22 nM T13260 C8I5JY 155511774 IC50 = 3200 nM T13260 C8ZYW2 155512683 Ki = 100 nM T13260 CWL61G 155513859 IC50 = 2750 nM T13260 COUZ40 155515111 Ki = 8 nM T13260 CQ0RX1 155519734 IC50 = 3300 nM T13260 CN8R0W 155521581 IC50 = 405 nM T13260 CS79RV 155522275 Ki = 24 nM T13260 CX9CY6 155523438 Ki = 97 nM T13260 C42DVB 155524075 Ki = 450 nM T13260 C7DX4M 155524253 IC50 = 110 nM T13260 CZCD39 155524316 Ki = 180 nM T13260 CO73MH 155528129 IC50 = 175 nM T13260 C9KHR3 155528792 IC50 = 210 nM T13260 C3PKZ1 155531378 IC50 = 0.2 nM T13260 CE2F1S 155532984 Ki = 81 nM T13260 C65EOC 155533109 Ki = 74 nM T13260 C2YTO1 155533392 IC50 = 520 nM T13260 C57SRY 155539404 IC50 = 105 nM T13260 CA01UF 155542148 IC50 = 210 nM T13260 C05WZC 155544203 Ki = 79 nM T13260 C1CJ3W 155544206 IC50 = 43.55 nM T13260 CZ48QO 155544544 IC50 = 660 nM T13260 C8NOR7 155548567 IC50 = 39.77 nM T13260 CO2G9W 155552576 IC50 = 73.17 nM T13260 C5CKA6 155553716 IC50 = 90.73 nM T13260 CAK73M 155557092 IC50 = 430 nM T13260 CA2H5K 155557102 IC50 = 17.42 nM T13260 C04ZVY 155557805 IC50 > 12500 nM T13260 CAY1Z7 155558257 IC50 = 14.52 nM T13260 CH3N8S 155558347 IC50 = 280 nM T13260 CJX17H 155558789 Ki = 57 nM T13260 CO6W0R 155559106 Ki = 125 nM T13260 C47PER 155559543 IC50 = 19.66 nM T13260 CH3IK5 155559681 IC50 = 8720 nM T13260 C3SWX8 155559867 IC50 = 58.85 nM T13260 CXT67R 155559873 IC50 = 560 nM T13260 CQU6N2 155562191 Ki = 290 nM T13260 C20AJK 155564333 IC50 = 55 nM T13260 CZ1OQ8 155569008 IC50 = 30.19 nM T13260 CH20CY 3114838 IC50 = 441 nM T13260 D00BVP 11847320 IC50 = 79.43 nM T13260 D00EMF 3644637 IC50 > 100000 nM T13260 D00HVZ 5271544 IC50 = 1860 nM T13260 D00RIX 5280443 IC50 = 1000 nM T13260 D00TWK 185914 IC50 > 50000 nM T13260 D00VUO 6539777 IC50 = 6360 nM T13260 D00ZPJ 408350 Ki = 25.5 nM T13260 D01IJX 10537337 IC50 = 3560 nM T13260 D01JZO 2779191 IC50 = 70 nM T13260 D01KKU 5281894 IC50 = 30.5 nM T13260 D01LOU 2238 IC50 = 40 nM T13260 D01MPK 12331302 Ki = 1750 nM T13260 D01REI 46901610 IC50 = 2440 nM T13260 D01SUE 6539759 IC50 = 2040 nM T13260 D01SZX 46867545 IC50 = 150 nM T13260 D01UYI 5281607 IC50 = 1 nM T13260 D02ALK 11514074 IC50 = 2700 nM T13260 D02BGR 9949648 IC50 = 13000 nM T13260 D02BWQ 6539818 IC50 = 2800 nM T13260 D02BXS 46901445 IC50 = 24560 nM T13260 D02CSU 6539786 IC50 = 12735030.81 nM T13260 D02LTV 10019821 IC50 = 110 nM T13260 D02LWB 6540046 IC50 > 36000 nM T13260 D02NAG 6539765 IC50 = 4260 nM T13260 D02QSH 339914 Ki = 1.9 nM T13260 D02SIT 9926623 IC50 = 74 nM T13260 D02XHH 6540043 IC50 = 100 nM T13260 D02XTS 6539811 IC50 = 3630 nM T13260 D03EXD 49864181 IC50 = 3070 nM T13260 D03FBI 49798900 IC50 = 8510 nM T13260 D03KLN 11413434 IC50 = 129 nM T13260 D03LOG 5280450 IC50 = 48000 nM T13260 D03MKT 6539788 IC50 = 1550 nM T13260 D03TRM 6540032 IC50 = 955 nM T13260 D03VRC 2989557 IC50 = 338.84 nM T13260 D04CLL 6539775 IC50 = 4720 nM T13260 D04DZZ 11646165 IC50 = 910 nM T13260 D04ELJ 6539766 IC50 = 4050 nM T13260 D04HVL 364705 IC50 = 2790 nM T13260 D04IBH 11616637 IC50 = 9107 nM T13260 D04IJE 256445 IC50 = 2741574.17 nM T13260 D04ISG 11680597 IC50 > 2000 nM T13260 D04LWL 97252 IC50 > 115600 nM T13260 D04QPK 6539783 IC50 = 1810 nM T13260 D04REX 6539808 IC50 = 790 nM T13260 D04TBB 10354739 IC50 = 2 nM T13260 D04VRY 11847169 IC50 = 467.74 nM T13260 D04WJN 10588478 IC50 = 389.05 nM T13260 D04ZGF 10561174 IC50 = 500 nM T13260 D05FFY 14231155 IC50 = 15 nM T13260 D05HBF 5353357 IC50 = 8.7 nM T13260 D05HRP 13596072 Ki = 800 nM T13260 D05IWY 5464078 IC50 = 4970 nM T13260 D05MQE 6539785 IC50 = 230 nM T13260 D05PXK 11847171 IC50 = 1800 nM T13260 D05QPR 12229388 IC50 = 880 nM T13260 D05YCI 42618032 IC50 = 18470 nM T13260 D05YJR 5495926 IC50 = 5200 nM T13260 D05YNW 6539790 IC50 = 6700 nM T13260 D05ZPO 1890 IC50 = 3800 nM T13260 D06AZC 135494055 IC50 = 1400 nM T13260 D06DDT 5315502 IC50 = 30000 nM T13260 D06FHE 44341253 IC50 = 205 nM T13260 D06GIV 337660 IC50 = 3100 nM T13260 D06HFV 6539805 IC50 = 7447319.74 nM T13260 D06HJB 14355826 IC50 = 55 nM T13260 D06PRC 5281650 IC50 = 20700 nM T13260 D06UQR 15306616 IC50 = 14800 nM T13260 D06WPP 11847170 IC50 = 4073.8 nM T13260 D07CTI 10853186 IC50 = 977.24 nM T13260 D07FGX 6116651 IC50 = 3300 nM T13260 D07IQG 10473365 IC50 = 933.25 nM T13260 D07JKK 11760063 IC50 = 1 nM T13260 D07LUJ 64945 IC50 = 14 ug.mL-1 T13260 D07PHT 324288 Ki = 6.5 nM T13260 D07PHV 10546089 IC50 = 89 nM T13260 D07PYC 6539760 IC50 = 3550 nM T13260 D07SOM 11847316 IC50 = 71 nM T13260 D07TIJ 3828439 IC50 = 2818.38 nM T13260 D07TUX 11230598 IC50 = 31622.78 nM T13260 D07UVN 6440384 IC50 = 3080 nM T13260 D07ZCD 6539804 IC50 = 1710 nM T13260 D07ZYL 6539797 IC50 = 3720 nM T13260 D08ARY 339906 Ki = 5.6 nM T13260 D08AZK 6539767 IC50 = 7830 nM T13260 D08EZA 11847317 IC50 = 45 nM T13260 D08FAB 11845485 IC50 > 2000 nM T13260 D08FHU 42618033 IC50 = 2720 nM T13260 D08FOJ 9898204 IC50 = 4300 nM T13260 D08HPU 6540052 IC50 = 1787 nM T13260 D08IIW 46887422 IC50 = 40 nM T13260 D08ISK 42618030 IC50 > 91290 nM T13260 D08KLN 13580711 IC50 = 3210 nM T13260 D08PKR 10845522 IC50 = 3060 nM T13260 D08PNF 6539770 IC50 = 5570 nM T13260 D08TKB 46889432 IC50 = 389.2 nM T13260 D08UQH 53600 IC50 = 190 nM T13260 D08ZTZ 11529133 IC50 = 1805 nM T13260 D09CPC 13728862 IC50 > 5000 nM T13260 D09DRS 42618031 IC50 = 960 nM T13260 D09HEA 1236449 IC50 = 1096.48 nM T13260 D09HGK 6539796 IC50 = 3960 nM T13260 D09HOE 6539789 IC50 = 800 nM T13260 D09HQH 13308 Ki = 260 nM T13260 D09MQF 15696376 IC50 = 900 nM T13260 D09MYQ 261365 Ki = 266 nM T13260 D09OPA 44593508 IC50 = 3400 nM T13260 D09QDY 6540033 IC50 = 130 nM T13260 D09TUB 11099375 IC50 > 308300 nM T13260 D09VPA 6539794 IC50 = 3400 nM T13260 D09VQM 442428 IC50 = 5000 nM T13260 D09XKH 10356745 IC50 = 2200 nM T13260 D09YXV 6539769 IC50 = 4310 nM T13260 D09ZHX 11847318 IC50 = 436.52 nM T13260 D09ZIW 10143276 IC50 = 7100 nM T13260 D0A0JL 2052 IC50 = 70600 nM T13260 D0A2FO 2825024 IC50 = 8000 nM T13260 D0A2GB 13660221 IC50 = 1300 nM T13260 D0A4EA 445639 IC50 = 32700 nM T13260 D0A4XA 25093379 IC50 > 50000 nM T13260 D0A7PA 49799639 IC50 = 11140 nM T13260 D0AH1B 6539782 IC50 = 12618275.35 nM T13260 D0AM2Z 13660216 IC50 = 11000 nM T13260 D0AW7Q 46867544 IC50 = 7900 nM T13260 D0AY4E 6539780 IC50 = 3930 nM T13260 D0B5MZ 13660218 IC50 = 2300 nM T13260 D0B8PE 10355761 IC50 = 3500 nM T13260 D0BH2T 10107266 IC50 > 40 ug.mL-1 T13260 D0C3XU 46887018 IC50 = 7 nM T13260 D0C5SV 5280934 IC50 = 44200 nM T13260 D0C5ZP 16125122 IC50 = 2140 nM T13260 D0C8EO 6539806 IC50 = 4330 nM T13260 D0C8KC 1504717 IC50 = 960 nM T13260 D0CR6B 11847319 IC50 = 69 nM T13260 D0D0DR 10081625 IC50 = 310 nM T13260 D0D7GG 510040 IC50 = 950 nM T13260 D0D8GU 6539803 IC50 = 1280 nM T13260 D0D8YE 6540048 IC50 = 5700 nM T13260 D0D9FR 6539795 IC50 = 3962780.34 nM T13260 D0DJ3R 10585323 IC50 = 100 nM T13260 D0DO1T 9819080 Ki = 10.3 nM T13260 D0DY5G 443389 IC50 > 100000 nM T13260 D0E2RV 360578 IC50 = 1700 nM T13260 D0E3IK 11680642 IC50 = 2510 nM T13260 D0E5FV 5318585 IC50 = 100 nM T13260 D0E9WX 6540042 IC50 = 27 nM T13260 D0F4MF 49799640 IC50 = 980 nM T13260 D0F4WQ 46867547 IC50 = 5.59 nM T13260 D0F5AC 46867542 IC50 = 17 nM T13260 D0F5YU 6539793 IC50 = 1990 nM T13260 D0F8IB 25256842 IC50 = 16500 nM T13260 D0F9MQ 11493409 IC50 = 2670 nM T13260 D0G2JV 49799657 IC50 = 2280 nM T13260 D0G6QL 23644748 IC50 = 2800 nM T13260 D0GL0L 11232117 IC50 = 3981.07 nM T13260 D0H1LK 161760 IC50 = 10200 nM T13260 D0HC9U 46867416 IC50 = 53 nM T13260 D0HD9P 444899 IC50 = 28200 nM T13260 D0HR9S 388623 Ki = 15.1 nM T13260 D0I1SI 49799655 IC50 = 760 nM T13260 D0I1YH 46901446 IC50 = 663 nM T13260 D0I2UE 46867543 IC50 = 3.98 nM T13260 D0I5NW 6540047 IC50 = 4073 nM T13260 D0I5PY 23585406 IC50 = 210 nM T13260 D0I7GE 11790 Ki = 20 nM T13260 D0J2WW 6539801 IC50 = 770 nM T13260 D0J3PK 11779089 IC50 = 41 nM T13260 D0J4VR 46191176 IC50 = 5000 nM T13260 D0J8FS 5377857 IC50 = 8330 nM T13260 D0JE1I 9815923 IC50 = 680 nM T13260 D0K2SE 10703161 IC50 = 6400 nM T13260 D0K3CE 6539800 IC50 = 280 nM T13260 D0K4PY 114829 IC50 = 2100 nM T13260 D0K5GG 49799652 IC50 = 3570 nM T13260 D0K5JU 46867417 IC50 = 1900 nM T13260 D0K5KG 6540050 IC50 = 6045 nM T13260 D0K8QD 63059 IC50 = 24880 nM T13260 D0L1JF 6539791 IC50 = 180 nM T13260 D0L3AJ 5324988 IC50 = 2020 nM T13260 D0L9BT 10823163 IC50 = 3700 nM T13260 D0M0FE 3317166 IC50 = 160 nM T13260 D0M2IB 9904788 Ki = 4 nM T13260 D0M4CX 356713 Ki = 385 nM T13260 D0M5EW 11276192 IC50 = 2089.3 nM T13260 D0M7FS 6539764 IC50 = 2490 nM T13260 D0M8RO 6128 Ki = 20 nM T13260 D0MA9G 6540051 IC50 = 1507 nM T13260 D0N1GH 11601068 IC50 > 36000 nM T13260 D0N1PQ 11506923 IC50 = 586 nM T13260 D0N5GZ 12229395 IC50 = 24500 nM T13260 D0N7QV 11819989 IC50 = 0.7 nM T13260 D0N9PY 6539773 IC50 = 7080 nM T13260 D0NB8V 49799650 IC50 = 16420 nM T13260 D0NH6T 14218027 IC50 = 400 nM T13260 D0NX0M 6540049 IC50 = 814 nM T13260 D0O0BL 44394887 IC50 = 430 nM T13260 D0O1ZM 13660225 IC50 = 1500 nM T13260 D0O4YS 42618026 IC50 > 98490 nM T13260 D0O6ZM 14256024 IC50 = 670 nM T13260 D0OY1J 11401873 IC50 = 676.08 nM T13260 D0P3ND 46887506 IC50 = 160 nM T13260 D0P5ZV 261861 IC50 = 9800 nM T13260 D0PU5V 10750911 IC50 = 1380 nM T13260 D0Q0BK 46901611 IC50 = 1670 nM T13260 D0Q3JZ 6539774 IC50 = 7680 nM T13260 D0Q6XB 5844100 IC50 = 7470 nM T13260 D0Q8UZ 18785180 IC50 = 590 nM T13260 D0QL1V 508445 IC50 = 1200 nM T13260 D0R0TE 11557864 IC50 = 6638 nM T13260 D0R2YN 5994480 IC50 = 15500 nM T13260 D0R4FM 122850 IC50 > 40 ug.mL-1 T13260 D0R4WW 44265823 Ki = 10.3 nM T13260 D0RJ6S 11558270 IC50 > 36000 nM T13260 D0S0EP 585819 IC50 = 28.18 nM T13260 D0S0OV 10267149 IC50 = 91 nM T13260 D0S0RK 10680 IC50 = 8 nM T13260 D0S1AY 269167 IC50 = 26800 nM T13260 D0S7VY 49798801 IC50 = 2940 nM T13260 D0S8MJ 337743 IC50 = 2100 nM T13260 D0S9YX 5280373 IC50 = 10.2 nM T13260 D0SY2M 5281708 Ki = 100000 nM T13260 D0SY6C 5282073 IC50 = 2 nM T13260 D0T0CK 49799648 IC50 = 14510 nM T13260 D0T3ED 44580826 Ki = 33.4 nM T13260 D0T3PW 5281672 IC50 = 10000 nM T13260 D0T5NO 15306617 IC50 = 100 nM T13260 D0TM4K 6539817 IC50 = 3680 nM T13260 D0U4BB 10748 IC50 > 10000 nM T13260 D0U6IT 6539807 IC50 = 4830 nM T13260 D0U6NJ 11311402 IC50 = 758.58 nM T13260 D0U7RR 6539768 IC50 = 7370 nM T13260 D0U8JC 9862769 IC50 = 4600 nM T13260 D0U9QB 73440 IC50 = 15 nM T13260 D0UI8Q 10566470 IC50 = 2089.3 nM T13260 D0V0DB 46887421 IC50 = 20 nM T13260 D0V1UY 133966 IC50 = 3 nM T13260 D0V3MV 46867546 IC50 = 11.45 nM T13260 D0V3YH 6539784 IC50 = 130 nM T13260 D0V8CR 6539763 IC50 = 2540 nM T13260 D0V8SM 10659706 IC50 = 1096.48 nM T13260 D0W3LG 9866908 IC50 = 9700 nM T13260 D0W3LM 10265122 IC50 = 3700 nM T13260 D0W4IB 23644623 Ki = 680 nM T13260 D0W7GU 5377410 IC50 = 1820 nM T13260 D0W7JA 5273567 IC50 = 35300 nM T13260 D0W9PF 13472 Ki = 43 nM T13260 D0W9ZC 46867540 IC50 = 16.5 nM T13260 D0WK9Q 14256034 IC50 = 2760 nM T13260 D0WN9P 46901444 IC50 = 2830 nM T13260 D0X0IH 77918 IC50 = 150 nM T13260 D0X1QS 6540053 IC50 = 3551 nM T13260 D0X8UK 10751574 IC50 = 350 nM T13260 D0XQ6T 42618029 IC50 = 5760 nM T13260 D0XS6T 53602 IC50 = 1840 nM T13260 D0Y0CT 6539819 IC50 = 4060 nM T13260 D0Y0EK 620596 IC50 = 3400 nM T13260 D0Y0QI 10774864 IC50 = 170 nM T13260 D0Y4TE 340000 Ki = 13.1 nM T13260 D0Y5KX 46901443 IC50 = 24500 nM T13260 D0Y7HG 5281616 Ki = 100000 nM T13260 D0Y7RB 6539781 IC50 = 4600 nM T13260 D0Y8XJ 5497182 IC50 = 16800 nM T13260 D0Y9HD 361928 Ki = 52.7 nM T13260 D0YD9J 6539792 IC50 = 5432503.31 nM T13260 D0YS2F 6539776 IC50 = 9740 nM T13260 D0Z1OI 124662 Ki = 1000 nM T13260 D0Z4GR 4594970 IC50 = 100 nM T13260 D0Z7EL 5280647 IC50 = 11000 nM T93509 D00MXN 25019940 Ki = 0.024 nM T93509 D0G5ME 11319053 Ki = 0.78 nM T93509 D0L5GH 6918509 Ki = 0.014 nM T93509 CXZA43 457930 Ki = 7300 nM T93509 C6W7AM 9847811 Ki = 2700 nM T93509 CANV26 10030220 Ki = 710 nM T93509 CH2NR6 11178760 Ki = 1700 nM T93509 C1LX9V 11397043 Ki = 1800 nM T93509 C8GB7A 11419496 Ki = 1900 nM T93509 CQT6I4 16728074 Ki = 16000 nM T93509 C5RC3J 44563430 IC50 >= 1000 nM T93509 C2BKH7 44563440 EC50 = 0.05 nM T93509 CQ1VU2 57392038 Ki = 26000 nM T93509 CF8R4H 57392039 Ki > 100000 nM T93509 C9T7IA 57393753 Ki = 8000 nM T93509 C6UID4 57393754 Ki = 5200 nM T93509 C1O0EL 57393755 Ki > 100000 nM T93509 C6B2JK 57395477 Ki = 14000 nM T93509 CD91MC 57395478 Ki = 45000 nM T93509 CV87FO 57397325 Ki > 100000 nM T93509 CK6L0F 57400721 Ki = 8 nM T93509 C6GF8M 57402496 Ki > 100000 nM T93509 CL85VH 57402497 IC50 > 10000 nM T93509 CPYG07 73345650 IC50 = 0.85 nM T93509 CH9LP4 73345651 IC50 = 3.45 nM T93509 CJ2V8U 73347156 IC50 = 29.73 nM T93509 C4DWG3 73347157 IC50 = 79.34 nM T93509 C8F9IO 73353230 IC50 = 4.15 nM T93509 CC5Q0Y 73354735 Ki = 0.73 nM T93509 CH7GY0 73354736 Ki = 3.3 nM T93509 C3LV6M 73356281 IC50 = 1.31 nM T93509 C3WJM4 127026899 IC50 = 130 nM T93509 CAJ24S 127026900 IC50 = 13 nM T93509 C7ZF6X 127026901 IC50 = 170 nM T93509 C6TRP3 127027478 IC50 = 15 nM T93509 C63EQW 127027479 IC50 = 19 nM T93509 C5VS7T 127027480 IC50 = 77 nM T93509 C26QAE 127027481 IC50 = 12 nM T93509 C9TR7O 127027482 IC50 = 22 nM T93509 C8DPY7 127027501 IC50 = 190 nM T93509 C1MW5C 127027502 IC50 = 460 nM T93509 CEK1B2 127027503 IC50 = 9.8 nM T93509 C9N5SC 127027797 IC50 = 44 nM T93509 C23NCY 127027803 IC50 = 33 nM T93509 C6JT4M 127027804 IC50 = 130 nM T93509 CXNT13 127027805 IC50 = 130 nM T93509 CI4Z3K 127027806 IC50 = 8.9 nM T93509 CZD67W 127027807 IC50 = 99 nM T93509 CR8GD0 127027810 IC50 = 110 nM T93509 CJH92D 127027811 IC50 = 44 nM T93509 C1BFU9 127027812 IC50 = 120 nM T93509 C0JIC7 127027814 IC50 = 350 nM T93509 CWS56B 127027815 IC50 = 4.3 nM T93509 CH0S6M 127027816 IC50 = 12 nM T93509 CQ3CR8 127027821 IC50 = 140 nM T93509 C0UGB6 127027822 IC50 = 97 nM T93509 CQ56CX 127027823 IC50 = 150 nM T93509 CT95NM 127027824 IC50 = 41 nM T93509 C3IJR5 127028113 IC50 = 46 nM T93509 CBJ5A4 127028116 IC50 = 7 nM T93509 C8SCZ7 127028121 IC50 = 34 nM T93509 CW1D3C 127028122 IC50 = 2.9 nM T93509 CDU86M 127028128 IC50 = 14 nM T93509 C1VEB4 127028129 IC50 = 0.23 nM T93509 CD70TW 127028130 IC50 = 0.11 nM T93509 C86NMZ 127028438 IC50 = 170 nM T93509 CHO8T2 127028443 IC50 = 92 nM T93509 C4Z1ND 127028444 IC50 = 120 nM T93509 CHM0F8 127028769 IC50 = 240 nM T93509 CM25XZ 127028770 IC50 = 54 nM T93509 C4NR9D 127028771 IC50 = 1.1 nM T93509 CTO2K3 127028772 IC50 = 19 nM T93509 CJ4IZ2 127028773 IC50 = 16 nM T93509 CPE3B1 127028774 IC50 = 24 nM T93509 CQ9R3C 127028775 IC50 = 430 nM T93509 D05LMD 16134896 Ki = 3.19 nM T93509 D0I2KW 44406785 IC50 = 740 nM T93509 D0U4BO 44563409 IC50 = 0.64 nM T08446 D0ED7U 60648 IC50 = 1670000 nM T08446 D08ESA 198693 IC50 = 300000 nM T08446 D0C9XA 119 IC50 = 2000 nM T08446 CJ9V4G 40598 IC50 = 290000 nM T08446 CXSD61 155246 IC50 = 3000 nM T08446 CHV0G9 639062 IC50 > 1000000 nM T08446 C97FYX 702501 IC50 = 100000 nM T08446 C8X9TQ 1069892 IC50 = 2884.03 nM T08446 C1A0UL 1502074 IC50 = 7943.28 nM T08446 C3DR8J 1502075 IC50 = 3981.07 nM T08446 C9EI4M 1530639 IC50 > 1000000 nM T08446 CU23IC 4531494 IC50 = 208000 nM T08446 CG1ZF6 5311322 Ki = 1600 nM T08446 CN2C7Q 6604883 IC50 = 630000 nM T08446 C4A6SU 8181355 IC50 = 180000 nM T08446 CQ64IH 9797818 IC50 = 7210000 nM T08446 C31HNE 9884272 Ki = 42000 nM T08446 CY2IS7 9888224 IC50 = 39000 nM T08446 CTZ5Q7 9983570 IC50 = 2660000 nM T08446 C75BDY 10031163 IC50 = 201000 nM T08446 CZ4PO2 10050339 IC50 = 1270000 nM T08446 CP2WF1 10072112 IC50 = 27000 nM T08446 CG1A4H 10073933 IC50 = 151000 nM T08446 C4S1CO 10096504 IC50 = 382000 nM T08446 C0XI3N 10252046 IC50 = 920000 nM T08446 CXJR61 10252950 IC50 = 655000 nM T08446 CC8V4E 10412575 IC50 = 109000 nM T08446 CZ8FQ2 10481573 IC50 = 88000 nM T08446 CU40KP 11743493 IC50 = 435000 nM T08446 CH6GX1 13314232 IC50 = 91000 nM T08446 C6VK4E 17173775 IC50 > 1000000 nM T08446 CE92MX 17174058 IC50 > 1000000 nM T08446 C3OQD7 17250318 IC50 = 170000 nM T08446 CME93B 43345728 IC50 > 1000000 nM T08446 C5JUW9 47058964 IC50 > 1000000 nM T08446 CLIK30 50941729 IC50 > 100000 nM T08446 CQ4XJ7 55285849 IC50 = 5480 nM T08446 CY9O8W 55285850 IC50 = 5480 nM T08446 C8UTR2 67642717 IC50 = 7300 nM T08446 C6ME5H 70684991 IC50 = 335000 nM T08446 C79CYX 70689234 IC50 = 2900000 nM T08446 CD9EV5 70691307 IC50 = 809000 nM T08446 CJ7P8C 70691309 IC50 = 436000 nM T08446 C53QGB 118711599 IC50 = 590 nM T08446 CO18BS 137635197 IC50 = 8000 nM T08446 CQL64H 137637846 IC50 > 1000000 nM T08446 CZ73DV 137638595 IC50 > 100000 nM T08446 CARI53 137638617 IC50 > 100000 nM T08446 CUM2T0 137638836 IC50 > 100000 nM T08446 C3PY5G 137638838 IC50 > 50000 nM T08446 CP7OV5 137639241 IC50 > 100000 nM T08446 C21IZT 137639281 IC50 > 1000000 nM T08446 CP24OX 137642163 IC50 > 100000 nM T08446 CK2VU3 137650102 IC50 > 1000000 nM T08446 C52PYO 137650910 IC50 > 1000000 nM T08446 CS6FX4 137651374 IC50 > 1000000 nM T08446 CPLJ94 137651669 IC50 > 1000000 nM T08446 CN04QK 137652511 IC50 > 1000000 nM T08446 CGC1Z4 137654858 IC50 > 50000 nM T08446 CADN74 137657292 IC50 > 100000 nM T08446 C4NK1W 137658990 IC50 > 50000 nM T08446 CPI4S8 137659917 IC50 > 50000 nM T08446 CI7S8H 155516242 IC50 > 100000 nM T08446 C4U8QT 155524561 IC50 > 100000 nM T08446 CJ4OV6 155530359 IC50 > 100000 nM T08446 C4RL9X 155535776 IC50 > 100000 nM T08446 CL2Q6G 155567178 IC50 > 100000 nM T08446 D02ANG 5216267 IC50 = 47400 nM T08446 D03IWW 6575389 IC50 = 6410000 nM T08446 D08YGM 92409 IC50 = 7210000 nM T08446 D0D2EF 1796510 IC50 = 2310000 nM T08446 D0H7WK 10458835 IC50 = 71700 nM T08446 D0P3KI 9888030 IC50 = 5100 nM T08446 D0RF2M 4498 IC50 = 2370000 nM T08446 D0V5OY 16725912 Ki = 15000 nM T08446 D0V7RG 3532 IC50 = 1870000 nM T97537 CQ5T2C 2837573 Ki = 7700 nM T97537 CIBH72 3834735 Ki > 100000 nM T97537 CA1ZC4 4188970 Ki = 5000 nM T97537 C4EBQ6 8823441 IC50 = 1100 nM T97537 CT45FK 24828324 Ki = 147.91 nM T97537 C1WKD6 24828325 Ki = 20.42 nM T97537 CJ6RS7 24828326 Ki = 5754.4 nM T97537 C98VUW 24828598 Ki = 5370.32 nM T97537 CW64AC 24828600 Ki = 144.54 nM T97537 CFP01R 24828743 Ki = 100 nM T97537 C9LUM1 24828881 Ki = 27.54 nM T97537 CER36P 24828882 Ki = 2137.96 nM T97537 C0VL7B 24890303 Ki = 10715.19 nM T97537 CJ6G0Y 42601512 Ki = 480 nM T97537 CL2A3I 42610322 Ki = 20 nM T97537 C12CDQ 44254309 Ki = 3019.95 nM T97537 C8EI1G 44254310 Ki = 8511.38 nM T97537 CD3L0N 44254402 Ki = 794.33 nM T97537 CHT0Z1 44254404 Ki = 2454.71 nM T97537 CW7LB9 44254495 Ki = 2041.74 nM T97537 C5FDC2 44254496 Ki = 2951.21 nM T97537 CE40ON 44277843 Ki = 52 nM T97537 CID3S9 44450222 Ki = 177.83 nM T97537 CCJ39L 44450246 Ki = 1071.52 nM T97537 CX05EH 44450286 Ki = 173.78 nM T97537 C87BVH 44450320 Ki = 165.96 nM T97537 C98XEN 44450334 Ki = 1318.26 nM T97537 CD7UO5 44450345 Ki = 630.96 nM T97537 CH02ZM 44450376 Ki = 81.28 nM T97537 CD85RG 44450377 Ki = 109.65 nM T97537 CZ4H7R 44560401 Ki = 1200 nM T97537 C70AIZ 44560402 Ki = 12000 nM T97537 C63VWA 44560403 Ki = 7400 nM T97537 CRX2G5 44560404 Ki = 2500 nM T97537 CA4IF6 44560405 Ki = 1400 nM T97537 C57LTE 44560406 Ki = 3700 nM T97537 C2F3TI 44560407 Ki = 3100 nM T97537 CC3GY2 44560408 Ki = 1300 nM T97537 C9YE7J 44560409 Ki = 1300 nM T97537 C1OEW5 44560410 Ki = 1800 nM T97537 CU4G1S 44560411 Ki = 1000 nM T97537 C2Y0OT 44560412 Ki = 97000 nM T97537 CG7BQ8 44560457 Ki = 16000 nM T97537 C1RK3C 44560557 Ki = 35000 nM T97537 C42VEQ 44560558 Ki = 76000 nM T97537 CMLG10 46882676 Ki = 4786.3 nM T97537 CTO1Q8 46882677 Ki = 3981.07 nM T97537 CP9WB0 49840768 Ki = 282 nM T97537 C51YRX 49840770 Ki = 54.8 nM T97537 CJ3Z7V 49840772 Ki = 1752 nM T97537 CS3I8G 49840774 Ki = 3.3 nM T97537 C3IT5V 49840844 Ki = 242 nM T97537 CYBW37 49840846 Ki = 18.5 nM T97537 CFEC23 49840848 Ki = 93.7 nM T97537 C64XMG 49840850 Ki = 5.2 nM T97537 CNU1Q7 49840921 Ki = 34.9 nM T97537 CQ90FE 52941108 Ki = 5506 nM T97537 CU4HK1 52943524 Ki = 196 nM T97537 C9HRG4 52946764 Ki = 22.5 nM T97537 C89EGH 52947188 Ki = 9.3 nM T97537 CU58OG 53257413 Ki = 4.1 nM T97537 C6XY5R 53259047 Ki = 50 nM T97537 C7AXD8 53259048 Ki = 41.1 nM T97537 CX51OK 53259216 Ki = 697 nM T97537 CBS92H 53259217 Ki = 351 nM T97537 C8RZW7 53259219 Ki = 5845 nM T97537 C4KZ7R 53259403 Ki = 4011 nM T97537 CA0Q2E 53259404 Ki = 12000 nM T97537 C6FU2G 53259405 Ki = 10800 nM T97537 CLSC37 53261358 Ki = 25 nM T97537 CXMC12 53261359 Ki = 64.2 nM T97537 C3Q4ZR 53261360 Ki = 193 nM T97537 CGF98A 54585162 Ki = 30.4 nM T97537 CG46AV 71817662 IC50 = 38300 nM T97537 C7P2UD 71817806 IC50 = 3900 nM T97537 CW85UH 71817807 IC50 > 100000 nM T97537 CO8K1H 71817808 IC50 = 46000 nM T97537 CMQN63 71817809 IC50 = 10300 nM T97537 CPNL07 71817811 IC50 = 9600 nM T97537 C1N7QD 71817963 IC50 = 2800 nM T97537 CMBJ36 71817964 IC50 = 1300 nM T97537 CK2T9X 71817965 IC50 = 16300 nM T97537 CE7VJ4 71817966 IC50 > 100000 nM T97537 C74CNV 72193911 IC50 = 30 nM T97537 C8ZGB7 118734158 IC50 = 10000 nM T97537 C0T8FC 118734159 IC50 = 10700 nM T97537 CU5F3O 118734160 IC50 = 57000 nM T97537 CB67XZ 118734161 IC50 = 10900 nM T97537 CJ19XY 118734162 IC50 = 2100 nM T97537 C67EIN 118734163 IC50 = 12000 nM T97537 C5HV4G 118734165 IC50 = 7200 nM T97537 CB7W1N 118734166 IC50 = 14600 nM T97537 CVQ9B5 118734167 IC50 = 34000 nM T97537 CTE28S 118734169 IC50 > 100000 nM T97537 C3VMB4 118734170 IC50 = 3800 nM T97537 C5B3AO 118734171 IC50 = 4800 nM T97537 CR02XN 118734172 IC50 = 10700 nM T97537 CYQ61P 118734173 IC50 = 5700 nM T97537 CG1NJ3 118734176 IC50 = 4100 nM T97537 CTL4C9 118734177 IC50 > 100000 nM T97537 CWK18R 118734179 IC50 = 12000 nM T97537 CED26H 118734180 IC50 > 100000 nM T97537 C24VOF 118734181 IC50 = 22000 nM T97537 C3KJR9 118734182 IC50 > 100000 nM T97537 CMWH70 118734252 IC50 = 7100 nM T97537 CS1R6T 118734253 IC50 > 100000 nM T97537 CK3NV4 118734254 IC50 = 933 nM T97537 C4VK6O 118734255 IC50 = 4400 nM T97537 C7AH4D 118734256 IC50 = 1300 nM T97537 CZ04FM 118734257 IC50 > 100000 nM T97537 CZ97HL 118734258 IC50 = 1200 nM T97537 C1DKP8 118734259 IC50 = 105 nM T97537 CET0D8 118734260 IC50 = 296 nM T97537 C4N7KF 118734261 IC50 = 31000 nM T97537 C2M4UZ 118734262 IC50 = 3300 nM T97537 C3PL1T 118734263 IC50 = 966 nM T97537 C3OS1H 118734264 IC50 = 655 nM T97537 C9NWC0 118734265 IC50 = 31000 nM T97537 C3PW9J 118734266 IC50 = 1700 nM T97537 CX0OA9 118734267 IC50 = 8300 nM T97537 CU8I4F 118734268 IC50 = 3300 nM T97537 CI6S8L 118734269 IC50 = 39600 nM T97537 C6IB5P 118734270 IC50 > 100000 nM T97537 CUGM56 118734271 IC50 = 9900 nM T97537 CH2LO8 118734272 IC50 = 22500 nM T97537 CI9RT3 118734273 IC50 > 100000 nM T97537 CK32TS 118734274 IC50 = 2500 nM T97537 CT5F3Q 118734275 IC50 = 20600 nM T97537 C3KLH4 118734276 IC50 = 14400 nM T97537 CPUI84 118734277 IC50 = 20200 nM T97537 C96PKA 118734278 IC50 = 1300 nM T97537 C4AL9Z 118734279 IC50 = 2400 nM T97537 C71TGN 118734280 IC50 = 4700 nM T97537 C8V9EB 118734281 IC50 = 2900 nM T97537 CIZ3Q6 118734282 IC50 = 3700 nM T97537 CJ64ZC 118734283 IC50 = 3800 nM T97537 C1K7AN 118734284 IC50 = 1300 nM T97537 C6XY9M 118734285 IC50 = 70000 nM T97537 CY8X0V 118734286 IC50 = 3400 nM T97537 CO4F3Y 118734287 IC50 = 5200 nM T97537 C9CN6S 118734288 IC50 = 3700 nM T97537 CI3R0S 118734289 IC50 > 100000 nM T97537 CN7SR4 118734290 IC50 = 3900 nM T97537 C57ZSG 118734291 IC50 > 100000 nM T97537 CKST54 118734292 IC50 = 3600 nM T97537 C9XDY5 118734293 IC50 = 438 nM T97537 C01PYL 118734294 IC50 = 1700 nM T97537 CO6PR7 118734295 IC50 = 35700 nM T97537 C4ZPC8 118734296 IC50 = 2200 nM T97537 CJ40TN 118734297 IC50 = 7600 nM T97537 CA9X0N 118734298 IC50 = 4900 nM T97537 C7FMV5 126456392 Ki = 18 nM T97537 C8QO7V 135554374 IC50 = 28000 nM T97537 CXLS30 137633011 IC50 = 381 nM T97537 CMC5E8 137634250 IC50 = 18 nM T97537 CER06G 137637900 IC50 = 577 nM T97537 C97XKO 137638141 IC50 = 16 nM T97537 CMTG53 137639983 IC50 = 1754 nM T97537 CH6DQ2 137640549 IC50 = 281 nM T97537 C9SWV7 137640590 IC50 = 46 nM T97537 CG0ED2 137641900 IC50 = 14 nM T97537 C3SP9K 137642894 IC50 = 317 nM T97537 C1U3ZM 137642974 IC50 = 1800 nM T97537 CYN9Z5 137646376 IC50 = 41 nM T97537 CDU93R 137646849 IC50 = 13 nM T97537 C96EWT 137647165 IC50 = 32 nM T97537 CJM57W 137648545 IC50 = 13 nM T97537 CC9T7O 137650040 IC50 = 9 nM T97537 CN9F2A 137650752 IC50 = 185 nM T97537 CB9VI7 137652734 IC50 = 102 nM T97537 CSM3V5 137653412 IC50 = 221 nM T97537 CVI87E 137654495 IC50 = 21 nM T97537 C8DV5C 137655020 IC50 = 4024 nM T97537 C2RIG6 137655030 IC50 = 4 nM T97537 CMT56C 137655972 IC50 = 434 nM T97537 C13POW 137656080 IC50 = 561 nM T97537 CCTK37 137657323 IC50 = 34 nM T97537 C4VS2D 137658289 IC50 = 20 nM T97537 CKHE71 137659752 IC50 = 10 nM T97537 C0ID7T 137660529 IC50 = 2 nM T97537 C8E6UD 137661774 IC50 = 29 nM T97537 CV2U0Z 137662110 IC50 = 41 nM T97537 D02MNM 71817810 IC50 = 6000 nM T97537 D04DTE 53259050 Ki = 1.8 nM T97537 D0L3PY 123814 Ki = 7 nM T88415 COQ0J9 9846486 IC50 = 3500 nM T88415 CSH73Q 43230121 IC50 = 5000 nM T88415 C09TSQ 145978898 IC50 = 100 nM T88415 CFX8E2 145979186 IC50 > 100000 nM T88415 CS9M7U 145990033 IC50 = 800 nM T88415 CS2HG5 145991728 IC50 = 100 nM T88415 C4K2YT 145992615 IC50 > 10000 nM T40488 D05VZE 119031 IC50 = 10000 nM T40488 D03BOZ 3342298 IC50 = 0.54 nM T40488 CN6E3U 2366268 IC50 = 83000 nM T40488 CR7T3J 10009978 Ki > 2000 nM T40488 C1LCH3 10016964 IC50 = 62000 nM T40488 CR5H6E 10163627 IC50 = 1600 nM T40488 CK0P3F 10186536 IC50 > 10000 nM T40488 C4K1MJ 10208262 IC50 = 4600 nM T40488 CBM0Y4 10252411 Ki < 100 nM T40488 CY08WJ 10322755 Ki = 1650 nM T40488 CFKA79 10395015 Ki > 2000 nM T40488 C5WV1N 10439082 Ki > 2000 nM T40488 C8C5AV 11294179 IC50 > 10000 nM T40488 CO8QT0 11753905 Ki = 240 nM T40488 C8YWV5 11778852 IC50 = 53000 nM T40488 C02BWA 11967143 Ki > 2000 nM T40488 CQS0F5 16719301 IC50 = 55 nM T40488 C75XDI 16730519 IC50 = 2400 nM T40488 C1MCG7 22004293 Ki = 335 nM T40488 CAQ9Z1 25022681 Ki > 5346 nM T40488 CHQG04 44576676 Ki = 23000 nM T40488 CR65DO 44576708 Ki = 1600 nM T40488 C2QFY7 44576710 Ki = 4570 nM T40488 CU2IP7 44576753 Ki = 22000 nM T40488 C93LDF 44576807 Ki = 372000 nM T40488 CJ41MB 44576851 Ki = 337000 nM T40488 CU2SX3 51355576 Ki > 10000 nM T40488 C6Y2EV 53374826 IC50 > 100000 nM T40488 C1PHI6 57708731 IC50 = 820 nM T40488 CF2Z7W 57708783 IC50 = 140 nM T40488 C9KV2W 57708792 IC50 = 460 nM T40488 CE36GP 57708799 IC50 = 270 nM T40488 C23QGY 57708843 IC50 > 1000 nM T40488 C2J5CW 57708880 IC50 > 1000 nM T40488 C1K6AP 57708886 IC50 = 30 nM T40488 C61NKZ 72720906 IC50 = 21 nM T40488 C7XWM5 72948626 IC50 = 17 nM T40488 CR70EY 72948808 IC50 = 12 nM T40488 C2WV4D 72948991 IC50 = 7810 nM T40488 CA76TR 72948995 IC50 = 18 nM T40488 CZ95GN 72949172 IC50 = 16 nM T40488 CSH7A5 90033597 IC50 = 11400 nM T40488 CYZP25 91824169 IC50 > 10000 nM T40488 C0M3QS 118179775 IC50 = 42 nM T40488 C0XML2 118179776 IC50 = 62 nM T40488 C0W3NG 118179777 IC50 = 435 nM T40488 CX9YG0 118179779 IC50 = 7 nM T40488 CW1TU9 118179786 IC50 = 54 nM T40488 CRG2W5 118179799 IC50 = 189 nM T40488 CH35NR 118179800 IC50 = 9 nM T40488 CK54UB 118179801 IC50 = 739 nM T40488 CP8QO0 118179807 IC50 = 13 nM T40488 CT4G5D 118179817 IC50 = 68 nM T40488 CIU02H 118179819 IC50 = 4 nM T40488 CD9TG2 118179830 IC50 = 103 nM T40488 CN72KV 118179833 IC50 = 184 nM T40488 CZ01AH 118179837 IC50 = 713 nM T40488 C6TR4O 118179845 IC50 = 25400 nM T40488 C5TZ1D 118179847 IC50 = 14 nM T40488 CVWR97 118179850 IC50 = 20700 nM T40488 CT8U1K 118179865 IC50 = 8700 nM T40488 CR64FW 118179867 IC50 = 84 nM T40488 CIXQ34 118179870 IC50 = 3 nM T40488 C27XIK 118225133 IC50 > 10000 nM T40488 C58KIN 118233723 IC50 > 10000 nM T40488 CU6ES2 118233724 IC50 > 10000 nM T40488 C8ET1Z 118233725 IC50 > 10000 nM T40488 C9P0LC 118233726 IC50 > 10000 nM T40488 C8SIM0 118233727 IC50 > 10000 nM T40488 CQTE52 118233728 IC50 > 10000 nM T40488 CEVI64 118233730 IC50 > 10000 nM T40488 C08CPE 118233731 IC50 > 10000 nM T40488 C8Q5XC 118233733 IC50 > 10000 nM T40488 CZQO42 118233734 IC50 > 10000 nM T40488 CCDG68 118233743 IC50 > 10000 nM T40488 C25TYU 118233744 IC50 > 10000 nM T40488 CL5UV6 118233745 IC50 > 10000 nM T40488 C8XWB9 118233746 IC50 > 10000 nM T40488 CC7K9R 118233747 IC50 > 10000 nM T40488 CGA7J1 118233748 IC50 > 10000 nM T40488 CVIG81 118233749 IC50 > 10000 nM T40488 CTU81Y 118233750 IC50 > 10000 nM T40488 CCA6W2 118233751 IC50 > 10000 nM T40488 C60QIZ 118233752 IC50 > 10000 nM T40488 CS5G9T 118233753 IC50 > 10000 nM T40488 CGKD16 118734983 IC50 = 32 nM T40488 C84NEC 118734984 IC50 = 89 nM T40488 CX7H5Q 118734985 IC50 = 17 nM T40488 CNF86U 121493953 Ki = 1.4 nM T40488 CH1GT7 123144081 IC50 > 10000 nM T40488 CKNI84 127050262 IC50 = 8400 nM T40488 CN9D7G 134155756 IC50 = 6300 nM T40488 CHV2U1 135438561 IC50 = 160 nM T40488 C6GR3K 135567051 IC50 = 140 nM T40488 CYH23I 136054468 IC50 = 220 nM T40488 CZ8DW1 136054472 IC50 = 34 nM T40488 C9H0DL 136054473 IC50 = 460 nM T40488 CX7MI0 136054475 IC50 = 64 nM T40488 CA5JR6 136054481 IC50 = 240 nM T40488 CO2VU9 136054484 IC50 < 10 nM T40488 CV47JN 136054485 IC50 = 6.2 nM T40488 CZ48WO 136054487 IC50 = 150 nM T40488 CR9CY5 136054490 IC50 < 10 nM T40488 C8FGT0 136054495 IC50 = 930 nM T40488 CGH39U 136054498 IC50 < 10 nM T40488 C2TO7Y 136054508 IC50 = 640 nM T40488 CG70BZ 136054516 IC50 = 0.35 nM T40488 CSM57W 136054520 IC50 = 2.6 nM T40488 CIEW62 136380958 IC50 = 2.4 nM T40488 C9HS7J 137287436 IC50 = 0.3 nM T40488 CAZ87R 137631621 IC50 = 676.08 nM T40488 C0R5ZT 137635841 IC50 = 436.52 nM T40488 CU5G8I 137636679 IC50 = 635 nM T40488 C1RID9 137636861 IC50 = 2050 nM T40488 CNM8J4 137638970 IC50 = 29.51 nM T40488 C7Y0FB 137642170 IC50 = 1210 nM T40488 CDOQ29 137644394 IC50 = 1698.24 nM T40488 C04KVQ 137647395 IC50 = 705 nM T40488 CHI2E1 137648744 IC50 = 112.2 nM T40488 C1U2QR 137651063 IC50 = 141.25 nM T40488 C5Y8RP 137654086 IC50 = 7380 nM T40488 CRD46H 137658344 IC50 = 347 nM T40488 C3ER5O 137658673 IC50 = 506 nM T40488 CEQ8I9 137659945 IC50 = 588.84 nM T40488 CHO70T 137660954 IC50 = 751 nM T40488 C1IF6L 137661809 IC50 = 131 nM T40488 CYFQ54 144883303 IC50 > 10000 nM T40488 CA2EI4 144883305 IC50 > 10000 nM T40488 CX80ML 144883318 IC50 > 10000 nM T40488 CQYH92 145949456 IC50 > 10000 nM T40488 C2SM0T 145950300 IC50 > 10000 nM T40488 C85BXD 145951133 IC50 > 10000 nM T40488 C6JP8O 145955500 IC50 > 10000 nM T40488 CXT3I5 145958912 IC50 > 10000 nM T40488 CQN59P 145959729 IC50 > 10000 nM T40488 CX6R5D 145959924 IC50 > 10000 nM T40488 C0K4JW 145972664 IC50 > 10000 nM T40488 CF64GH 155518335 Ki = 983 nM T40488 D03AMR 9849669 Ki = 190 nM T40488 D04VPH 45376872 IC50 = 16000 nM T40488 D07SPC 24857837 Ki = 356 nM T40488 D0B3UN 44580458 Ki = 149 nM T40488 D0OR6O 91623362 IC50 = 12 nM T40488 D0Y5IQ 44255320 IC50 = 5000 nM T10877 D04AIT 5280445 IC50 = 8200 nM T10877 D0K8KX 5280343 IC50 = 37900 nM T10877 D0E3LP 5113032 IC50 > 100000 nM T10877 D0U3EP 445154 IC50 > 100000 nM T10877 CU12QE 1203 IC50 > 100000 nM T10877 CEM9Q1 128853 IC50 = 14600 nM T10877 CNMW58 159287 IC50 = 17000 nM T10877 CAB1I4 440832 IC50 = 16300 nM T10877 CT2S6P 441667 IC50 = 6300 nM T10877 CG5OR9 441697 IC50 = 14200 nM T10877 CHE81U 441701 IC50 = 6000 nM T10877 CXB75J 441773 IC50 = 20900 nM T10877 CXG1I8 441774 IC50 = 39200 nM T10877 CLY6K3 661302 IC50 > 100000 nM T10877 CJ0T4E 3612016 IC50 > 100000 nM T10877 CY9C4T 5281680 IC50 = 48600 nM T10877 C4KG0A 5403988 IC50 = 296000 nM T10877 CKC79O 10053069 IC50 = 276000 nM T10877 C5J6HV 11170346 IC50 = 158000 nM T10877 CU7Y3S 12309895 IC50 = 70300 nM T10877 C5VH6T 14842007 IC50 = 32100 nM T10877 C4DQJ9 24285123 IC50 = 120000 nM T10877 C36ILR 44532635 IC50 = 1210 nM T10877 CLX72I 59474759 IC50 > 30000 nM T10877 C5GB8X 91827499 IC50 = 76 nM T10877 C64QCZ 91827500 IC50 = 7200 nM T10877 CM01EG 101886781 IC50 = 27000 nM T10877 CWC1Q3 101886782 IC50 = 6400 nM T10877 C5G1LT 101886783 IC50 = 33000 nM T10877 CDT01C 101886784 IC50 = 3300 nM T10877 CQUF15 118736849 IC50 = 58 nM T10877 C5KPU3 118736852 Ki = 14 nM T10877 CG7I6Z 118736853 IC50 = 52 nM T10877 CDR8M7 118736855 IC50 = 3.9 nM T10877 C3M6IP 118736856 Ki = 0.3 nM T10877 CZSB48 118736857 Ki = 0.7 nM T10877 CIE3W9 118736858 IC50 = 54 nM T10877 CH26AO 118736859 IC50 = 3.8 nM T10877 CAQM69 118736860 IC50 = 13 nM T10877 CEL48B 118736861 Ki = 0.45 nM T10877 C7JQ3Y 118736862 IC50 = 14 nM T10877 C6MZ9V 118736863 IC50 = 10773 nM T10877 C0U5DA 118736864 IC50 = 498 nM T10877 CZVT62 118736865 IC50 = 959 nM T10877 CE21BJ 118736866 IC50 = 1960 nM T10877 C30BIV 118736867 IC50 = 11400 nM T10877 CC10IV 118736868 IC50 = 3350 nM T10877 CXO8F1 118736869 IC50 = 2300 nM T10877 CAYX13 118736870 IC50 = 23400 nM T10877 CDW94Q 118736871 IC50 > 30200 nM T10877 CY4LA6 118736872 IC50 = 4710 nM T10877 CTCH72 118736873 IC50 = 1160 nM T10877 C3ARY5 118736874 IC50 = 1590 nM T10877 CW4O7N 118736875 IC50 = 263 nM T10877 CL51QY 118736876 IC50 = 206 nM T10877 CKMD80 118736877 IC50 = 28 nM T10877 CY93JQ 118736878 IC50 = 26 nM T10877 C73EMV 118736879 IC50 = 64 nM T10877 C1B2JZ 118736880 IC50 = 53 nM T10877 C5KGR7 118736881 IC50 = 42 nM T10877 CVM02C 118736882 IC50 = 245 nM T10877 CCH64S 118736883 IC50 = 50 nM T10877 CB6S3J 118736884 IC50 = 3.4 nM T10877 C2SWZ4 118736886 IC50 = 4.8 nM T10877 CXEC56 118736887 IC50 = 5.3 nM T10877 C9LJ0B 118736888 IC50 = 298 nM T10877 C06HDY 118736889 IC50 = 840 nM T10877 CT8G1K 118736890 IC50 = 1200 nM T10877 CUN41C 118736891 IC50 = 1320 nM T10877 CGJW47 118736892 IC50 = 700 nM T10877 CAU39P 118736893 IC50 = 3610 nM T10877 CT5A7R 118736894 IC50 = 2330 nM T10877 C1YMX6 118736895 IC50 = 970 nM T10877 C0RD2H 118736896 IC50 = 4680 nM T10877 CO70TW 118736897 IC50 = 1230 nM T10877 C8HC3W 118736898 IC50 = 1160 nM T10877 CK2LV7 118736899 IC50 = 12800 nM T10877 CXQ37E 118736900 IC50 = 2150 nM T10877 CRT50V 118736901 IC50 = 700 nM T10877 CPAE18 118736902 IC50 = 970 nM T10877 CUPZ76 118736903 IC50 = 2690 nM T10877 CA87UE 118736904 IC50 = 560 nM T10877 CS59UX 118736905 IC50 = 840 nM T10877 CL7CR9 118736906 IC50 = 460 nM T10877 CT0EM6 118736907 IC50 = 1460 nM T10877 C3AJ1K 118736908 IC50 = 12300 nM T10877 CXJQ24 118736909 IC50 = 3940 nM T10877 CL0OQ1 118736910 IC50 = 950 nM T10877 C8TWX1 118736911 IC50 = 7830 nM T10877 C4OW8Z 118736912 IC50 = 1930 nM T10877 C6W4EN 118736913 IC50 = 281 nM T10877 C4FY6U 118736914 IC50 = 132 nM T10877 C6M7KH 118736915 IC50 = 1680 nM T10877 C3U9ZQ 118736916 IC50 = 1060 nM T10877 CN3DE6 118736989 IC50 = 1030 nM T10877 C3A5TU 118736990 IC50 > 30200 nM T10877 C7USD5 118736991 IC50 > 30200 nM T10877 CH1XL4 118736992 IC50 = 149 nM T10877 C2U9HL 118736993 IC50 = 1220 nM T10877 CI24RE 118736994 IC50 = 117 nM T10877 CDC8E7 118736995 IC50 = 140 nM T10877 CND2U1 118736996 IC50 = 49 nM T10877 C1BGP6 118736997 IC50 = 142 nM T10877 CMO4B9 118736998 IC50 = 406 nM T10877 C0Y4VE 118736999 IC50 = 78 nM T10877 CDV30H 118737000 IC50 = 971 nM T10877 C0XI5O 118737001 IC50 = 92 nM T10877 CQD48J 122185943 IC50 > 30000 nM T10877 C6Y2MI 122185944 IC50 = 22000 nM T10877 CR9G7S 122185945 IC50 = 22000 nM T10877 CD64IJ 122185946 IC50 = 3300 nM T10877 CE9OP1 122185947 IC50 > 30000 nM T10877 CBEL62 122185948 IC50 > 30000 nM T10877 CYM8D4 122185949 IC50 = 19000 nM T10877 CE1ZO9 122185950 IC50 > 30000 nM T10877 CE6VJ3 122185951 IC50 > 30000 nM T10877 CX76QZ 122185952 IC50 = 17000 nM T10877 CZ8N9B 122185953 IC50 = 25000 nM T10877 CHE12L 122185954 IC50 = 3300 nM T10877 CL94EM 122185955 IC50 = 2300 nM T10877 CJ17HX 122185956 IC50 > 30000 nM T10877 CI01XG 122185957 IC50 = 18000 nM T10877 CR9AX0 122185958 IC50 = 620 nM T10877 C79BPI 122185959 IC50 > 30000 nM T10877 CZL15G 122185960 IC50 = 4500 nM T10877 CJOV10 122185961 IC50 > 30000 nM T10877 CY2W1Z 122185962 IC50 = 11000 nM T10877 CEV6S8 122185963 IC50 = 990 nM T10877 CM9A0O 122185964 IC50 > 30000 nM T10877 C6D9YZ 122185965 IC50 = 15000 nM T10877 C9CA8T 122185966 IC50 > 30000 nM T10877 C9KAB4 122185967 IC50 > 30000 nM T10877 CLJ1R3 122185968 IC50 = 16000 nM T10877 C6OA7C 122185969 IC50 = 4000 nM T10877 CH16FN 122185970 IC50 = 9600 nM T10877 C8V0WI 122185971 IC50 = 24000 nM T10877 C1FB8D 122185972 IC50 = 6200 nM T10877 CX89LW 122185973 IC50 = 780 nM T10877 CK0UN1 122185974 IC50 = 1200 nM T10877 CQ1WJ8 122185975 IC50 = 510 nM T10877 CKD43Z 122185976 IC50 = 150 nM T10877 CV73WF 122185977 IC50 = 4700 nM T10877 CS7YJ2 122185978 IC50 = 170 nM T10877 CEIT53 122185979 IC50 = 3600 nM T10877 C3ZNU8 122185980 IC50 = 130 nM T10877 CN5P3Q 122185981 IC50 = 280 nM T10877 CIU0M2 122185982 IC50 = 8500 nM T10877 C13TYI 122185983 IC50 = 7300 nM T10877 CSZ0K1 122185984 IC50 > 30000 nM T10877 C8OL5C 122185985 IC50 = 2100 nM T10877 CU47TS 122185986 IC50 = 4900 nM T10877 CVUP84 122185987 IC50 > 30000 nM T10877 CM47OU 122185988 IC50 = 11000 nM T10877 C1DVY8 122185989 IC50 > 30000 nM T10877 CI01VG 122185990 IC50 > 30000 nM T10877 C0M9EL 122185991 IC50 > 30000 nM T10877 CM4S0B 122185992 IC50 > 30000 nM T10877 CO2R4W 122185993 IC50 = 6600 nM T10877 CN4B2Y 122185994 IC50 = 2700 nM T10877 C8WPN3 122185995 IC50 > 30000 nM T10877 CUG8B4 122185996 IC50 > 30000 nM T10877 COYI82 122185997 IC50 > 30000 nM T10877 CSC4B7 122185998 IC50 > 30000 nM T10877 CSOI57 122185999 IC50 = 24000 nM T10877 CGAB47 122186000 IC50 > 10000 nM T10877 CB2H6L 122186001 IC50 > 30000 nM T10877 CZ3R6F 122186002 IC50 > 30000 nM T10877 C6DN9H 122186003 IC50 > 30000 nM T10877 CD0QV5 122186004 IC50 > 30000 nM T10877 CEHN13 122186005 IC50 > 30000 nM T10877 CKFD41 122186006 IC50 > 30000 nM T10877 CU87NS 122186007 IC50 > 30000 nM T10877 CSZ5T7 122186008 IC50 > 30000 nM T10877 C5DU6F 122186009 IC50 > 30000 nM T10877 CQB19L 122186010 IC50 = 9200 nM T10877 C46EGM 135900947 IC50 = 430000 nM T10877 C61OBZ 135949782 IC50 = 103000 nM T10877 C6MF7P 136124133 IC50 = 109000 nM T10877 C0E3AH 136198640 IC50 = 14000 nM T10877 CACG84 136198641 IC50 = 26000 nM T10877 C4Z1WR 137442659 IC50 = 1900 nM T10877 CN09RB 137442681 IC50 = 450 nM T10877 C9G6IA 137442708 IC50 = 630 nM T10877 C9PUZ4 137442715 IC50 = 620 nM T10877 C7DP2S 137442862 IC50 = 92 nM T10877 CW8LT6 137442987 IC50 = 2300 nM T10877 CK26ZH 145967624 IC50 = 7.8 nM T10877 C0YGC8 145967690 IC50 = 1600 nM T10877 CV90MY 145967850 IC50 = 110 nM T10877 C0KJD1 145967861 IC50 = 21 nM T10877 COYK91 145968096 IC50 = 370 nM T10877 CC4P8J 145968138 IC50 = 72 nM T10877 CIW3B1 145968359 IC50 = 3400 nM T10877 C6F4SD 145968563 IC50 = 4100 nM T10877 COA4B0 145968763 IC50 = 170 nM T10877 CX4GA2 145968779 IC50 = 310 nM T10877 C9YRW1 145968807 IC50 = 1900 nM T10877 C4D1JT 145968829 IC50 = 8000 nM T10877 C9SV6Y 145969196 IC50 = 17 nM T10877 CS70GC 145969309 IC50 = 82 nM T10877 CNH7O5 145969326 IC50 = 51 nM T10877 CHZ7N3 145969706 IC50 = 42 nM T10877 CN56YO 145969928 IC50 = 330 nM T10877 C4CDN0 145969972 IC50 = 83 nM T10877 C1I3TK 145970025 IC50 = 6800 nM T10877 C6A0HJ 145970175 IC50 = 140 nM T10877 CJC43R 145970183 IC50 = 5500 nM T10877 CMKZ95 145970214 IC50 = 4200 nM T10877 CB2NU1 145970392 IC50 = 1600 nM T10877 CJR21T 145970400 IC50 = 410 nM T10877 CQ82EI 145970446 IC50 = 4300 nM T10877 CORE90 145970461 IC50 = 230 nM T10877 C4GR7E 145970630 IC50 = 71 nM T10877 CB4RP9 145970636 IC50 = 160 nM T10877 C3LD1Y 145970800 IC50 = 20 nM T10877 C7N2ZY 145970856 IC50 = 45 nM T10877 CUSO84 145970885 IC50 = 110 nM T10877 CKDZ10 145971093 IC50 = 19000 nM T10877 CW6ER8 145987053 IC50 = 4 nM T10877 CYT73F 145987735 IC50 = 2500 nM T10877 D07NAY 5281692 IC50 = 37900 nM T10877 D0E1QP 4262314 IC50 > 100000 nM T10877 D0O0VZ 667639 IC50 > 100000 nM T10877 D0T3PW 5281672 IC50 = 24800 nM T10877 D0V3PG 128861 IC50 = 21800 nM T69912 D0T9TJ 3034010 IC50 = 50 nM T69912 D05GZD 9918381 IC50 = 0.2512 nM T69912 D0CW8S 71657619 IC50 > 10000 nM T69912 D09NBM 10417440 Ki = 0.03 nM T69912 D0L5UO 9939609 IC50 = 0.035 nM T69912 CN1K3D 5699 IC50 > 100000 nM T69912 CZI2U1 6491 IC50 > 1000000 nM T69912 CYFU26 130606 IC50 > 100000 nM T69912 CZ3R1F 669158 IC50 = 1000000 nM T69912 C2KRB1 973435 IC50 = 44000 nM T69912 CMN1P8 1217803 IC50 = 3431 nM T69912 C2F7OG 2412772 IC50 = 1000000 nM T69912 C9VZ3F 3638243 IC50 > 100000 nM T69912 C1FHP8 4811752 IC50 = 14000 nM T69912 CG0F8O 9808838 IC50 = 1 nM T69912 CC5Y0A 9809899 IC50 = 533 nM T69912 C4TB5Y 9831072 IC50 = 0.6 nM T69912 C4VH8G 9840384 IC50 = 850 nM T69912 CB0EP8 9850883 IC50 = 26 nM T69912 C4R6CU 9851531 IC50 = 20 nM T69912 C89RJZ 9852438 IC50 = 0.5 nM T69912 CTJO81 9893629 IC50 = 85 nM T69912 C9FWY2 9895919 IC50 = 2 nM T69912 C6MD8O 9917136 IC50 = 8 nM T69912 C19SKN 9917325 IC50 = 0.7 nM T69912 CX23UG 9917667 IC50 = 9 nM T69912 CMBO57 9917750 IC50 = 0.4 nM T69912 CSB71L 9938151 IC50 = 18 nM T69912 CFH61N 9938577 IC50 = 26 nM T69912 CMN74S 9938642 IC50 = 12 nM T69912 CGL13H 9939495 IC50 = 0.4 nM T69912 C2EF8Q 9939518 IC50 = 2 nM T69912 CQEN19 9959703 IC50 = 24 nM T69912 C8C0HB 9961561 IC50 = 1 nM T69912 CSW8T3 9961700 IC50 = 0.3 nM T69912 C8X7KP 9961715 IC50 = 9 nM T69912 C1DB0X 10055750 IC50 = 0.17 nM T69912 C1TY3F 10122289 IC50 = 0.25 nM T69912 C0KOC5 10122452 IC50 = 3 nM T69912 C1LSI8 10122657 IC50 = 0.1 nM T69912 CJ4R2U 10168216 IC50 = 0.4 nM T69912 CAK3E1 10189993 IC50 = 0.8 nM T69912 CPG87K 10189998 IC50 = 38 nM T69912 CG65NB 10190629 IC50 = 1 nM T69912 CIK7C8 10211722 IC50 = 1.5 nM T69912 CA4EF3 10211894 IC50 = 2 nM T69912 CFQ5L2 10232552 IC50 = 5 nM T69912 CB72SI 10233112 IC50 = 1 nM T69912 C9UIX5 10233517 IC50 = 0.8 nM T69912 C61ZEV 10282620 IC50 = 1 nM T69912 CQV98P 10305047 IC50 = 0.5 nM T69912 COAR34 10305066 IC50 = 19 nM T69912 CZA96C 10305422 IC50 = 0.8 nM T69912 C7W2NF 10305573 IC50 = 1 nM T69912 C8OPC6 10305637 IC50 = 6 nM T69912 C03CJA 10320992 IC50 = 64 nM T69912 C0JB9D 10394633 IC50 = 0.7 nM T69912 CD3MH2 10411777 IC50 = 54 nM T69912 CU78FP 11521655 IC50 = 25000 nM T69912 CZRT87 11543912 IC50 = 38000 nM T69912 CJW8M7 11564757 IC50 = 26000 nM T69912 C09ASJ 11764593 IC50 = 0.2 nM T69912 CU0Y2Z 12051594 IC50 = 2 nM T69912 C6O8ID 14490158 IC50 = 1000000 nM T69912 CS5CV2 16126765 IC50 = 120 nM T69912 CGN9S6 17899989 IC50 = 640 nM T69912 CK14ET 17899991 IC50 = 210 nM T69912 C8C4LK 18470089 IC50 = 110 nM T69912 C0EU2T 18470090 IC50 = 0.3 nM T69912 C63DZQ 18470117 IC50 = 19 nM T69912 C7FV0Y 18470125 IC50 = 850 nM T69912 CRS63W 18470138 IC50 = 90 nM T69912 CJ0Q9T 18470140 IC50 = 17000 nM T69912 CFI50Y 18470152 IC50 = 34 nM T69912 C1WJ5A 18470163 IC50 = 1000 nM T69912 CZJ25E 18470168 IC50 = 19 nM T69912 CK47RM 18470169 IC50 = 200 nM T69912 C69SCV 18470191 IC50 = 4 nM T69912 C38OXW 18470208 IC50 = 1400 nM T69912 C68IDK 18470209 IC50 = 1000 nM T69912 CYF0B8 18470218 IC50 = 4400 nM T69912 C24HOS 18470241 IC50 = 2 nM T69912 C1Q8NP 18470244 IC50 = 11 nM T69912 CIEQ59 18470251 IC50 = 780 nM T69912 CE69PL 18470253 IC50 = 210 nM T69912 CP5S1M 18470258 IC50 = 650 nM T69912 C1NLE8 18470267 Ki = 41 nM T69912 CA38TG 18470272 IC50 = 430 nM T69912 C9Z0PI 18470273 IC50 = 660 nM T69912 CUTF18 18470282 IC50 = 12000 nM T69912 C9BRG5 18470283 IC50 = 250 nM T69912 CBZ1V0 18470296 IC50 = 12600 nM T69912 CT10SU 18470303 IC50 = 19 nM T69912 CJ35LB 18470304 IC50 = 4400 nM T69912 CV2Q4O 18470306 IC50 = 150 nM T69912 C2EGW7 18470314 IC50 = 16 nM T69912 C6CVW9 18470315 IC50 = 7 nM T69912 CR6S2P 18470316 IC50 = 1300 nM T69912 CT1G0Z 18470322 IC50 = 285 nM T69912 CU3QI1 18470341 IC50 = 960 nM T69912 CEIF53 18470354 IC50 = 450 nM T69912 CS93WA 18470361 IC50 = 2900 nM T69912 C0BE4O 18470368 IC50 = 110 nM T69912 CLS52M 18470371 IC50 = 1000 nM T69912 C8HNR6 18470375 IC50 = 450 nM T69912 C7VK9N 18470385 IC50 = 300 nM T69912 CX6EC7 18470390 IC50 = 250 nM T69912 C45GTM 18470395 IC50 = 0.1 nM T69912 C2EL5G 18470399 IC50 = 55000 nM T69912 C60DVF 18470400 IC50 = 1200 nM T69912 CXW4D9 18470406 IC50 = 200 nM T69912 C07FGB 18470420 IC50 = 330 nM T69912 CPE8J7 18470422 IC50 = 5700 nM T69912 CE1Y8Q 18470432 IC50 = 1400 nM T69912 CL0GA7 18470436 IC50 = 1200 nM T69912 CUA07V 18470440 IC50 = 1100 nM T69912 C0TQ3E 18470452 IC50 = 1100 nM T69912 C5GC2U 18470455 IC50 = 1 nM T69912 CHN74T 18470468 IC50 = 70 nM T69912 C15KXN 18470470 IC50 = 2 nM T69912 CLGR76 18470474 IC50 = 2300 nM T69912 C14IMQ 18470482 IC50 = 630 nM T69912 CR50VA 18470483 IC50 = 1100 nM T69912 C78SLA 18470487 IC50 = 39 nM T69912 CDY3G7 18470494 IC50 = 230 nM T69912 CMFK89 18470498 IC50 = 36 nM T69912 CPI0Y6 18470516 IC50 = 250 nM T69912 CV47NE 18470522 IC50 = 110 nM T69912 C0FYD2 18470524 IC50 = 1100 nM T69912 CG18YS 18470527 IC50 = 7 nM T69912 CI9JK7 18470549 IC50 = 14000 nM T69912 C8Y9TC 18470552 IC50 = 140 nM T69912 CE83XT 18470555 IC50 = 3300 nM T69912 CJY4G6 18470556 IC50 = 1100 nM T69912 COIL12 18470582 IC50 = 2850 nM T69912 C1QV9I 18470585 IC50 = 990 nM T69912 CB95IU 18470590 IC50 = 0.4 nM T69912 CD2G1X 18470595 IC50 = 780 nM T69912 CH63UY 18540820 IC50 = 1 nM T69912 CRC64I 18768423 IC50 = 52.4 nM T69912 CY4AF7 21936103 IC50 = 0.1 nM T69912 C4VY5P 21936114 IC50 = 4 nM T69912 CMS86P 21936124 IC50 = 0.5 nM T69912 CDT3Y6 21936140 IC50 = 0.3 nM T69912 COEI56 21936146 IC50 = 5 nM T69912 C9C3JG 21936169 IC50 = 1 nM T69912 CN5ZP0 21936176 IC50 = 1 nM T69912 C4P8MH 21936183 IC50 = 0.2 nM T69912 C8U3FQ 21936197 IC50 = 8 nM T69912 C9PUJ0 21936206 IC50 = 15 nM T69912 CMR0P1 21936209 IC50 = 5 nM T69912 CB1W0U 21936229 IC50 = 4 nM T69912 CM8NF3 21936243 IC50 = 0.8 nM T69912 CV49NU 21936282 IC50 = 0.6 nM T69912 C6JX0D 21936319 IC50 = 0.2 nM T69912 CCU98M 21936326 IC50 = 3 nM T69912 CB5M3Q 21936345 IC50 = 0.2 nM T69912 CV8QT9 21936398 IC50 = 0.2 nM T69912 C0B2MU 21936403 IC50 = 4 nM T69912 CA4X5J 21936407 IC50 = 5 nM T69912 CEC2B6 22294074 IC50 = 0.5 nM T69912 C2BJY9 23395723 IC50 = 1 nM T69912 CW7FL6 23395729 IC50 = 0.6 nM T69912 C3CZL1 23395731 IC50 = 2.7 nM T69912 C02MBF 23395732 IC50 = 17 nM T69912 CDH5N2 23395748 IC50 = 8 nM T69912 C6Y9DO 23395749 IC50 = 4 nM T69912 CH3RP0 23395766 IC50 = 2 nM T69912 C0G8KF 23395772 IC50 = 0.7 nM T69912 C79IXE 23395774 IC50 = 0.12 nM T69912 CMQ2X3 23395778 IC50 = 1 nM T69912 CH7S9G 23395784 IC50 = 1.6 nM T69912 CXP67J 23395785 IC50 = 0.6 nM T69912 CFN51M 23395786 IC50 = 4.5 nM T69912 CVM86Y 23395788 IC50 = 1.4 nM T69912 C32CYB 23395790 IC50 = 0.8 nM T69912 C8A9OF 23395792 IC50 = 2 nM T69912 C4PL8S 23395794 IC50 = 5 nM T69912 CL2CM7 23395795 IC50 = 1 nM T69912 CW9G8Y 23395798 IC50 = 5 nM T69912 CE1J3W 23395801 IC50 = 0.7 nM T69912 CNDH71 23395803 IC50 = 0.2 nM T69912 CV9H3P 23395804 IC50 = 0.12 nM T69912 CH0G9B 23395805 IC50 = 0.2 nM T69912 CUXA85 23395806 IC50 = 0.35 nM T69912 C01DHS 23395807 IC50 = 0.5 nM T69912 CU2J0M 23395808 IC50 = 0.2 nM T69912 CET9J2 23395809 IC50 = 1.5 nM T69912 C73WNR 44266749 IC50 = 50 nM T69912 C4XW9G 44266800 IC50 = 3 nM T69912 C6OWG4 44300071 IC50 = 34 nM T69912 CKU80A 44300072 IC50 = 21 nM T69912 CLU67B 44300088 IC50 = 97 nM T69912 CD41MI 44300109 IC50 = 140 nM T69912 C6LK3F 44300123 IC50 = 66 nM T69912 C4CG6Q 44300126 IC50 = 1280 nM T69912 C1HYF9 44300132 IC50 = 460 nM T69912 CJE5Y8 44300187 IC50 = 39 nM T69912 CZ6M8X 44300263 IC50 = 350 nM T69912 CHR95L 44300266 IC50 = 260 nM T69912 C72MUZ 44300268 IC50 = 51 nM T69912 CZS4T9 44300303 IC50 = 44 nM T69912 CKNC02 44300306 IC50 = 70 nM T69912 C3WJC0 44300307 IC50 = 29 nM T69912 CUB07K 44300374 IC50 = 3 nM T69912 CD02LG 44300390 IC50 = 410 nM T69912 CQ7M6U 44300414 IC50 = 89 nM T69912 C3FAV2 44300418 IC50 = 6700 nM T69912 CX56UK 44300444 IC50 = 530 nM T69912 C8HPB9 44300446 IC50 = 720 nM T69912 C34HVB 44300478 IC50 = 130 nM T69912 C01MXK 44300573 IC50 = 10 nM T69912 CI2EA3 44300574 IC50 = 69 nM T69912 CK4D5X 44300578 IC50 = 5 nM T69912 CG5HW3 44300752 IC50 = 120 nM T69912 CXQI32 44300753 IC50 = 176 nM T69912 C4ZDS7 44319598 IC50 = 235 nM T69912 CVYP89 44319686 IC50 = 12 nM T69912 CFJD61 44319860 IC50 = 350 nM T69912 CH1TP7 44319861 IC50 = 300 nM T69912 CUV80P 44319972 IC50 = 250 nM T69912 COD96J 44319974 IC50 = 25 nM T69912 CJBU28 44319998 IC50 = 260 nM T69912 CCU1J0 44320037 IC50 = 3 nM T69912 C9UZM1 44320070 IC50 = 15 nM T69912 CL2A8D 44367433 IC50 = 1.6 nM T69912 C0BM7X 44367434 IC50 = 0.5 nM T69912 C0CNE9 44367483 IC50 = 1.6 nM T69912 C8HM0C 44367519 IC50 = 0.2 nM T69912 CGS4E6 44367542 IC50 = 1.7 nM T69912 C04WGR 44367559 IC50 = 5 nM T69912 C0Q9NA 44367560 IC50 = 2.6 nM T69912 CG7AQ0 44367583 IC50 = 0.9 nM T69912 CVB27E 44367645 IC50 = 194 nM T69912 CNK0A7 44367647 IC50 = 5 nM T69912 CQ6S3B 44367648 IC50 = 24 nM T69912 CP2GU1 53299144 IC50 > 100000 nM T69912 CCR5A9 56927662 IC50 = 59 nM T69912 CAG1J5 56927666 IC50 = 23 nM T69912 C6GKE8 56950525 IC50 = 16 nM T69912 C21HQB 57336782 IC50 = 3.4 nM T69912 C5WQ8S 57392555 IC50 = 96 nM T69912 CITS38 57394279 IC50 = 170 nM T69912 CR8GA1 57396026 IC50 = 31 nM T69912 CKN4Q7 57396027 IC50 = 55 nM T69912 C83CEW 57397828 IC50 = 64 nM T69912 CX65FQ 57397830 IC50 = 92 nM T69912 C89RKP 57397831 IC50 = 56 nM T69912 CN5L8A 57397832 IC50 = 91 nM T69912 CMBI04 57397833 IC50 = 2900 nM T69912 CK2C8H 57401254 IC50 = 61 nM T69912 CN9TM3 57401255 IC50 = 130 nM T69912 C4PC1W 57402997 IC50 = 4100 nM T69912 CF23GK 57402999 IC50 = 48 nM T69912 C5SE6Y 57403000 IC50 = 360 nM T69912 CLQ5P8 59900388 IC50 = 1 nM T69912 CL0FU7 63334771 IC50 = 100000 nM T69912 C59VAN 71181474 IC50 = 0.55 nM T69912 C13KJW 71181477 IC50 = 0.23 nM T69912 CI1Y9Z 71181626 IC50 = 1.6 nM T69912 CPXJ23 71181632 IC50 = 0.96 nM T69912 CML2I0 71181668 IC50 = 0.24 nM T69912 CU8YK1 71181747 IC50 = 1.72 nM T69912 C9B7MX 71181764 IC50 = 0.91 nM T69912 CO7K5M 71181859 IC50 = 0.46 nM T69912 C1FGZ5 71181861 IC50 = 0.81 nM T69912 CBG0P3 71181874 IC50 = 0.89 nM T69912 CO0W1H 71476859 IC50 = 0.14 nM T69912 CJPF24 71486715 IC50 = 0.86 nM T69912 C9DA6W 71562486 IC50 = 14000 nM T69912 C40WLD 71562487 IC50 = 230 nM T69912 C0N4SW 71562488 IC50 = 55 nM T69912 CS41XO 71562489 IC50 = 38 nM T69912 CB8E0O 71562597 IC50 = 370 nM T69912 CU02DS 71562598 IC50 = 86000 nM T69912 CX62RJ 71562599 IC50 = 820 nM T69912 CH5GA2 71562600 IC50 = 29000 nM T69912 C2XRB6 71562601 IC50 = 32 nM T69912 CL0KT3 71562602 IC50 = 9700 nM T69912 C6N7RZ 71562603 IC50 = 100 nM T69912 CT64JI 71562727 IC50 = 150 nM T69912 C8AOX0 71562728 IC50 = 150 nM T69912 CRX2Q4 71562729 IC50 = 16 nM T69912 CMWV34 71562730 IC50 = 70 nM T69912 CU4Z2Q 71562731 IC50 = 87 nM T69912 CJU1L8 71562732 IC50 = 44 nM T69912 CQ4AN0 71562733 IC50 = 240 nM T69912 CN15BR 71562848 IC50 = 3000 nM T69912 CY37JA 71562849 IC50 = 41000 nM T69912 C7APK1 71562850 IC50 = 31 nM T69912 CA1C8N 71562851 IC50 = 26 nM T69912 C4OBN3 71562852 IC50 = 13 nM T69912 C6PQG5 71562853 IC50 = 14 nM T69912 C50DMA 71562854 IC50 = 39 nM T69912 CCK65O 71562973 IC50 = 49 nM T69912 CUW2X3 71562974 IC50 = 52 nM T69912 CU2K4F 71562975 IC50 = 120 nM T69912 C1YI9V 71562976 IC50 = 250 nM T69912 C80IKC 71562977 IC50 = 450 nM T69912 CZEX42 71562978 IC50 = 100 nM T69912 C0TQ5W 71562979 IC50 = 39 nM T69912 CO8XE5 71563093 IC50 = 26 nM T69912 C71VWC 71563094 IC50 = 4 nM T69912 C42RMU 71563095 IC50 = 55 nM T69912 CQ39RC 71563096 IC50 = 28 nM T69912 CJU20T 71563097 IC50 = 3 nM T69912 CDJ92S 71563098 IC50 = 3 nM T69912 CUO97N 71563099 IC50 = 80 nM T69912 CC3LF8 71563229 IC50 = 22 nM T69912 C6G8OV 71614098 IC50 = 0.67 nM T69912 CPQ5H2 71614498 IC50 = 0.95 nM T69912 CYO64A 71656315 IC50 > 1000 nM T69912 C50OAM 71656796 IC50 = 210 nM T69912 C2TO5C 71656797 IC50 > 10000 nM T69912 CN89IX 71656798 IC50 = 93 nM T69912 C49OFR 71656799 IC50 = 26 nM T69912 C92YGU 71657082 IC50 = 5000 nM T69912 CV5PM2 71657185 IC50 = 10000 nM T69912 CPT0H5 71657290 IC50 = 10000 nM T69912 CM2ZB8 71657292 IC50 = 810 nM T69912 CBSW63 71657395 IC50 > 10000 nM T69912 CVUD47 71657398 IC50 > 10000 nM T69912 CV24SL 71716432 IC50 = 4 nM T69912 CTH15K 71717661 IC50 = 23 nM T69912 C1AYH2 71718263 IC50 = 32 nM T69912 CTPL54 71718264 IC50 > 100000 nM T69912 CS7WK3 74889411 IC50 > 100 nM T69912 C2KHF7 89677087 IC50 = 1400 nM T69912 CXT5C7 89682527 IC50 = 1500 nM T69912 CPF01Q 89682653 IC50 = 580 nM T69912 CY7PD2 89682704 IC50 = 930 nM T69912 CNU8L7 89682719 IC50 = 1800 nM T69912 C2JS9A 119057479 IC50 = 500000 nM T69912 CZL6P8 119057480 IC50 = 230 nM T69912 C1S6CA 119057481 IC50 = 2000 nM T69912 CV8MY3 119057482 IC50 = 1700 nM T69912 CGN2X5 119057483 IC50 = 230 nM T69912 CW6T2I 121005813 IC50 = 1.7 nM T69912 CL70DK 121448333 IC50 = 8.3 nM T69912 C3N6DK 121448334 IC50 = 1.8 nM T69912 CM4S9R 121448337 IC50 = 4.2 nM T69912 C9U7WD 121448368 IC50 = 1.6 nM T69912 CI86GD 121448372 IC50 = 1.9 nM T69912 C1A5GV 121448374 IC50 = 2.2 nM T69912 CKM5Z4 121448380 IC50 = 2.7 nM T69912 CW0V2U 121448402 IC50 = 4 nM T69912 CG9H1O 121448406 IC50 = 3.7 nM T69912 CRE5L4 121448411 IC50 = 2.2 nM T69912 CF65PJ 121448417 IC50 = 2.6 nM T69912 CX1LF9 121448418 IC50 = 8 nM T69912 C3OBQ9 121448429 IC50 = 4.6 nM T69912 CJ4F7G 121448430 IC50 = 1.2 nM T69912 CZM7L3 121448431 IC50 = 3.5 nM T69912 CSCG90 121448433 IC50 = 1.8 nM T69912 C8TVD7 121448459 IC50 = 1.1 nM T69912 COU74T 121448460 IC50 = 3.9 nM T69912 CIW92J 122196130 IC50 = 11.1 nM T69912 CY4XR8 122196132 IC50 = 10.6 nM T69912 CIY90U 122196137 IC50 = 19.3 nM T69912 C5AFS0 122196138 IC50 = 16 nM T69912 C32FMN 122196204 IC50 = 13.4 nM T69912 CJGP91 122196205 IC50 = 16.9 nM T69912 CKA4Y1 122196208 IC50 = 3.7 nM T69912 CCWJ26 122196209 IC50 = 2.9 nM T69912 C9WZI8 122196212 IC50 = 2.3 nM T69912 CEL90A 122196214 IC50 = 6.5 nM T69912 CQBA39 122196215 IC50 = 10.9 nM T69912 CI3CW8 122196216 IC50 = 6.3 nM T69912 C7JU5Q 122530045 IC50 = 6300 nM T69912 C5BW4Z 122707116 IC50 = 15000 nM T69912 CX92RI 122707117 IC50 = 1600 nM T69912 C23EKP 122707118 IC50 = 1000 nM T69912 CU95PT 122707120 IC50 = 32 nM T69912 CK05FL 127050954 IC50 = 3.6 nM T69912 C8TUI5 127050955 IC50 = 2.4 nM T69912 C7DA4S 127050956 IC50 = 18 nM T69912 C01RCH 127050977 IC50 = 30000 nM T69912 CJW7D2 127051244 IC50 = 560 nM T69912 C1GSK5 127053040 IC50 = 180 nM T69912 CRC6Z1 127053472 IC50 = 1.1 nM T69912 CU0D3S 130346049 IC50 = 1400 nM T69912 CH7EL8 132427687 IC50 = 14 nM T69912 CW74SC 134133758 IC50 = 75 nM T69912 CM5R6E 134135433 IC50 = 10000 nM T69912 CYXB84 134136689 IC50 = 39000 nM T69912 CM98WH 134137624 IC50 = 7900 nM T69912 C1SP0U 134138704 IC50 = 620 nM T69912 CJG9M7 134140857 IC50 = 1500 nM T69912 CP3HL5 134143019 IC50 = 860 nM T69912 CFQ13X 134144083 IC50 = 2700 nM T69912 C1GZ9U 134145078 IC50 = 2000 nM T69912 CUV5B0 134145387 IC50 = 5400 nM T69912 CSN0D4 134146496 IC50 = 1900 nM T69912 C5YD1G 134147073 IC50 = 6200 nM T69912 C8WF9X 134147739 IC50 = 20000 nM T69912 C69BXV 134148543 IC50 = 160 nM T69912 CCE7M2 134150004 IC50 = 0.3981 nM T69912 C36ZHN 134150110 IC50 = 11000 nM T69912 CXV2M9 134150242 IC50 = 4300 nM T69912 C58MQS 134152799 IC50 = 110 nM T69912 C8MA0Z 134153116 IC50 = 980 nM T69912 CZGB70 134154962 IC50 = 160 nM T69912 CA85UF 134155224 IC50 = 86 nM T69912 C16NSU 134155260 IC50 = 660 nM T69912 CHL74N 134156788 IC50 = 10000 nM T69912 CEW49V 134157408 IC50 = 72 nM T69912 C3SVZ5 134693749 IC50 = 355 nM T69912 C3DE5Y 134693750 IC50 = 5 nM T69912 CZ3F5D 135239539 IC50 = 844 nM T69912 C0U9TO 137546866 IC50 = 430 nM T69912 CH4MR3 137633945 IC50 = 902 nM T69912 CTD75A 137633962 IC50 = 9 nM T69912 CRCU09 137634263 IC50 = 236 nM T69912 CH05MV 137636050 IC50 = 613 nM T69912 CG3K6U 137637253 IC50 = 12 nM T69912 CMNT10 137638920 IC50 = 23 nM T69912 CK70BJ 137641309 IC50 = 42 nM T69912 C6LIG7 137642017 IC50 = 222 nM T69912 CZ3F7X 137642755 IC50 = 2477 nM T69912 CJP45C 137643198 IC50 = 924 nM T69912 CS4W0J 137643921 IC50 = 13 nM T69912 CA50JV 137645485 IC50 = 1027 nM T69912 C4F5GR 137647910 IC50 = 322 nM T69912 CFL68S 137649687 IC50 = 1070 nM T69912 CL61YI 137651817 IC50 = 152 nM T69912 CX3AJ9 137652098 IC50 = 17 nM T69912 CJ73YS 137654141 IC50 = 65 nM T69912 CSR0J2 137655061 IC50 = 57 nM T69912 CGBL78 137655982 IC50 = 232 nM T69912 CTU98S 137658155 IC50 = 100 nM T69912 C9X3WS 137658880 IC50 = 1915 nM T69912 CLVM39 137660910 IC50 = 45 nM T69912 C4JV2G 137661511 IC50 = 1418 nM T69912 CO67DI 137661556 IC50 = 45 nM T69912 CEQ7G4 155510849 IC50 > 10000 nM T69912 C9CD3Q 155511585 IC50 = 430 nM T69912 C25OAR 155512542 IC50 = 2000 nM T69912 CI2WL8 155513853 IC50 > 1000 nM T69912 CBG4Q8 155521008 IC50 > 1000 nM T69912 CL6Z1R 155526799 IC50 = 750 nM T69912 CW7N6K 155533489 IC50 = 1000 nM T69912 CQ67EK 155543660 IC50 = 1800 nM T69912 C8XZ7V 155545255 IC50 = 330 nM T69912 C9WGK1 155547201 IC50 = 1300 nM T69912 CH78YM 155549832 IC50 > 1000 nM T69912 C4U9WO 155550747 IC50 = 10000 nM T69912 D05LXG 5063 IC50 = 11000 nM T69912 D09QHC 7370 IC50 > 1000000 nM T69912 D0A1SO 11206881 IC50 = 3800 nM T69912 D0D7AS 11701397 IC50 = 11200 nM T69912 D0FO2B 1923 IC50 > 100000 nM T69912 D0JI8S 11470979 IC50 = 2000 nM T69912 D0WW7A 9939109 IC50 = 8 nM T69912 D0X6UV 11368513 IC50 = 4400 nM T89826 D04AIT 5280445 IC50 = 20000 nM T89826 D07EXH 359 IC50 > 200000 nM T89826 D07MGA 72281 IC50 = 8300 nM T89826 D0J9ZR 4477 IC50 = 40000 nM T89826 D0K8KX 5280343 IC50 = 8100 nM T89826 C5H9TY 14697 IC50 = 207000 nM T89826 C3I7VB 102678 IC50 = 24500 nM T89826 CL5Y4J 159516 Ki = 3100 nM T89826 CV0B7W 442027 IC50 = 49600 nM T89826 C1E2FR 442048 IC50 = 283500 nM T89826 CZ3MD8 647122 IC50 = 16100 nM T89826 C2C8QU 948801 Ki = 27500 nM T89826 CXA4P6 1265413 IC50 = 90720 nM T89826 CUD4A1 1328543 IC50 = 58350 nM T89826 C3ZP4U 2131972 Ki = 9110 nM T89826 CA1N3H 2131982 Ki = 9930 nM T89826 CKL8B2 2219105 IC50 = 29900 nM T89826 CN43XQ 2806068 IC50 = 160 nM T89826 C5J6MO 2849659 IC50 = 28800 nM T89826 CN3P7A 2911959 IC50 = 74500 nM T89826 CZDG23 2947583 IC50 = 186000 nM T89826 CBIP72 2986413 IC50 = 76700 nM T89826 CCU3P7 3635406 IC50 = 2200 nM T89826 CZF0R5 4004950 IC50 = 500 nM T89826 C3AN7C 4117477 IC50 = 1180 nM T89826 CS2WB7 4236803 IC50 = 29800 nM T89826 C0AW3N 4378077 IC50 = 13860 nM T89826 CO3Y0T 4614896 IC50 = 9910 nM T89826 CY68ZT 4788586 IC50 = 940 nM T89826 CTR4Q1 5320532 IC50 = 13300 nM T89826 CVG47I 5958938 IC50 = 10500 nM T89826 CD8ZT2 6026688 IC50 > 50000 nM T89826 C3LZX9 8027611 IC50 = 12660 nM T89826 CJ4C5K 9180583 IC50 = 10800 nM T89826 CYQ8Z4 9882716 IC50 > 50000 nM T89826 C8K2NO 10062715 IC50 = 800000 nM T89826 C49CMU 10411574 IC50 = 21700 nM T89826 C6GN2F 11642725 IC50 = 870000 nM T89826 CHYP53 12310492 IC50 = 233400 nM T89826 C65EOH 15949840 IC50 = 7500 nM T89826 C9V8EM 15956553 IC50 = 300000 nM T89826 C3WYR4 16061499 IC50 = 2000 nM T89826 CTO43V 16085283 Ki = 116000 nM T89826 CU35DQ 21582568 IC50 = 220800 nM T89826 CN45FL 23427055 IC50 = 164700 nM T89826 CK3AF8 25256829 IC50 = 5400 nM T89826 C2SZ7L 42624533 IC50 = 14000 nM T89826 CYP8V1 44404067 IC50 > 50000 nM T89826 CD20PF 44433696 IC50 = 80000 nM T89826 CI4P2V 44433697 IC50 = 10000 nM T89826 CW7B0J 44433698 IC50 = 15000 nM T89826 C8DWL3 44433699 IC50 = 200000 nM T89826 C0ZPE2 44517748 IC50 = 2700 nM T89826 C0OH2T 44584893 IC50 = 5400 nM T89826 C0NZ5E 44584944 IC50 = 7300 nM T89826 CT70DZ 44590821 IC50 = 22500 nM T89826 C0SW2K 45266425 IC50 = 2500 nM T89826 C5WBP2 45266482 IC50 = 3800 nM T89826 CA4K8F 45266488 IC50 = 6600 nM T89826 C3BHZ4 45268445 IC50 > 50000 nM T89826 CC05NI 45268452 IC50 = 15400 nM T89826 C6QD9E 45269292 IC50 > 50000 nM T89826 CY7RV4 45269761 Ki = 21000 nM T89826 CO80TH 45269762 Ki = 297000 nM T89826 CU34ZK 45269763 Ki = 584000 nM T89826 C9P3LZ 45269764 Ki = 478000 nM T89826 CXS19V 45269765 Ki = 45200 nM T89826 C3DY4T 45270971 IC50 > 50000 nM T89826 CR4WA8 45270979 IC50 = 20900 nM T89826 CM78GO 45271412 Ki = 462000 nM T89826 CC90BU 45271826 IC50 = 5200 nM T89826 C0B6KX 45271831 IC50 = 9300 nM T89826 CN85IQ 45271832 IC50 = 8100 nM T89826 C7IF2O 45272299 Ki = 363000 nM T89826 CZRV73 45272304 Ki = 34100 nM T89826 CGV14L 45272305 Ki = 112000 nM T89826 CVTL97 45272306 Ki = 2200 nM T89826 CAM89I 45273174 Ki = 135000 nM T89826 CZT67B 45273179 Ki = 614000 nM T89826 CHF4M5 45273180 Ki = 49300 nM T89826 CND1R3 45273184 Ki = 159000 nM T89826 C0V5WT 45273625 IC50 > 50000 nM T89826 C6OE7V 46784066 IC50 = 28300 nM T89826 C6LH5I 46881919 Ki = 800 nM T89826 CI2FO1 49870840 IC50 = 5500 nM T89826 CF2D0I 49870841 IC50 = 8400 nM T89826 CM52SZ 49870842 IC50 = 6800 nM T89826 C8Q2CZ 50885062 IC50 > 50000 nM T89826 CJ6KV7 52941131 IC50 = 13900 nM T89826 C8M2QD 52943127 IC50 = 24300 nM T89826 CQ84MD 52945913 IC50 = 12000 nM T89826 CJ1LG2 52945915 IC50 = 42000 nM T89826 CZ35DX 52945977 IC50 = 128900 nM T89826 CAB1Y3 52946772 IC50 = 163200 nM T89826 CO4R1B 52947200 IC50 = 18000 nM T89826 CC4X1O 52948928 IC50 = 137700 nM T89826 CMG4U7 52949213 IC50 = 10800 nM T89826 C0X5BL 58589722 IC50 = 76740 nM T89826 CY3CL6 71544384 IC50 = 610 nM T89826 CV3P2U 71544385 IC50 = 230 nM T89826 CJS60O 71571220 IC50 = 49000 nM T89826 C1AY0M 71571221 IC50 = 49000 nM T89826 CY21XB 71571222 IC50 = 4600 nM T89826 C1DX9H 71571223 IC50 = 39000 nM T89826 CKE2C3 73056463 IC50 > 100000 nM T89826 C9S8ZH 73056464 IC50 > 100000 nM T89826 CK9OI0 73056465 IC50 = 31710 nM T89826 C4D8LK 73056466 IC50 = 32080 nM T89826 CRY86G 73056467 IC50 = 34910 nM T89826 C3VS4F 73056760 IC50 = 10070 nM T89826 CYH1F4 73056761 IC50 = 51330 nM T89826 C2CRZ8 73056762 IC50 = 2250 nM T89826 CD4YR3 73056763 IC50 = 11830 nM T89826 C3P2OZ 73056764 IC50 = 67200 nM T89826 C1H8PX 73056765 IC50 = 82910 nM T89826 C8JO7B 73056766 IC50 = 13860 nM T89826 CCYE63 73057087 IC50 = 5520 nM T89826 C54JWM 73057088 IC50 = 39870 nM T89826 C8RBU6 73057089 IC50 = 1040 nM T89826 CEBH65 73057090 IC50 = 1690 nM T89826 C8M2DX 73057091 IC50 = 17820 nM T89826 CQ42AZ 73057092 IC50 = 2820 nM T89826 CPLJ64 73057388 IC50 = 4700 nM T89826 CIN5V0 76320984 IC50 = 4300 nM T89826 C05AYV 102341658 IC50 = 16400 nM T89826 C8S3CR 102341659 IC50 = 37500 nM T89826 C2G9CP 127043455 IC50 = 20200 nM T89826 CVZ4I3 127043641 IC50 = 6000 nM T89826 C7BST4 127043642 IC50 = 5800 nM T89826 CGO01F 127043643 IC50 > 50000 nM T89826 C2TU5A 127043644 IC50 = 6400 nM T89826 C0Y9IT 127043645 IC50 = 41200 nM T89826 CF3B1Z 127045220 IC50 = 11700 nM T89826 CIXJ94 127045221 IC50 = 8600 nM T89826 CQ1CT5 127045222 IC50 = 18700 nM T89826 CKRX04 127045227 IC50 = 30700 nM T89826 CDZ2E1 127045228 IC50 > 50000 nM T89826 CG3E9B 127045229 IC50 = 6700 nM T89826 CG6VR3 127045386 IC50 = 15700 nM T89826 CK9JE3 127045387 IC50 > 50000 nM T89826 CY1E4Z 127045392 IC50 > 50000 nM T89826 CK5PA4 127045393 IC50 = 44700 nM T89826 C34TWD 127045394 IC50 > 50000 nM T89826 C97MQC 127048409 IC50 = 20000 nM T89826 C41VRM 127048410 IC50 = 7500 nM T89826 CZ0B1R 127052510 IC50 = 10000 nM T89826 CRW05E 127052511 IC50 > 50000 nM T89826 CC3TX0 127052512 Ki = 72000 nM T89826 CIQ1U9 127052513 Ki = 41000 nM T89826 CI13JZ 135452883 IC50 = 10000 nM T89826 CG1KW5 135470831 IC50 = 77090 nM T89826 CH4Q6A 145964401 IC50 = 5500 nM T89826 CHU61S 145964420 IC50 = 42100 nM T89826 C6YCA8 145964710 IC50 = 28800 nM T89826 CV6F7L 145966788 IC50 = 2100 nM T89826 CBWX17 145967285 IC50 = 4300 nM T89826 COR9X3 145972736 IC50 = 3900 nM T89826 CQ0M2X 145972809 IC50 = 4100 nM T89826 CF95RZ 145972878 IC50 = 3200 nM T89826 CXI0D1 145975081 IC50 = 6300 nM T89826 CG84ZR 145975487 IC50 = 5100 nM T89826 C91FOT 145976006 IC50 = 5200 nM T89826 C3F4UH 145978039 IC50 = 8800 nM T89826 CL7FB0 2919450 IC50 = 62790 nM T89826 D00RIX 5280443 IC50 = 280800 nM T89826 D01XMM 4117383 IC50 = 4450 nM T89826 D08MZY 145937 Ki = 8200 nM T89826 D08UYP 3008868 Ki = 2400 nM T89826 D09BUG 10207 IC50 = 132000 nM T89826 D0L7AT 10480940 Ki = 19300 nM T89826 D0S0BN 130976 Ki = 10600 nM T89826 D0SY2M 5281708 IC50 = 105000 nM T89826 D0UQ6U 10569 IC50 = 189100 nM T89826 D0WA9S 10429214 IC50 = 146500 nM T90961 C3VRO9 44557921 IC50 > 10000 nM T90961 C67OJG 44588117 Ki = 4400 nM T90961 C4YWO9 134812845 Ki = 17 nM T90961 CG15PY 134812846 Ki > 100000 nM T90961 C9O8CQ 137348448 Ki = 13 nM T90961 C63TGO 137349551 Ki = 17 nM T90961 C6I5ME 137349552 Ki = 19 nM T90961 CRC8D2 155489850 Ki = 95000 nM T90961 CG8J5X 155518911 Ki = 27 nM T90961 CAN08J 155534113 Ki = 36 nM T90961 C16JRL 155535406 Ki = 74 nM T90961 C3XR8O 155536206 Ki = 51 nM T90961 CX68YN 155541385 Ki > 100000 nM T90961 CWU67H 155543077 Ki = 59 nM T90961 CD8K3O 155543384 Ki = 42 nM T90961 CUTW39 155546618 Ki = 20 nM T90961 C4E0HB 155546757 Ki = 120 nM T90961 C49UVQ 155547733 Ki = 17 nM T90961 CI2J4O 155551330 Ki = 37 nM T90961 CP2K8O 155554487 Ki = 30 nM T90961 CS8MC1 155562025 Ki = 33 nM T90961 C8UW4P 155562878 Ki = 17 nM T90961 CDP94M 155569521 Ki = 53 nM T88806 D0BN9X 60947 IC50 > 300000 nM T88806 D01TJY 53340771 IC50 = 7.7 nM T88806 D09ZXO 176873 IC50 = 13.2 nM T88806 D0Q5LF 9961766 IC50 > 100000 nM T88806 D08LIG 153986 IC50 > 3 nM T88806 D0P8JX 177831 IC50 > 5 nM T88806 C7CL3Y 107775 IC50 = 2200 nM T88806 CE19HD 132605 IC50 = 27000 nM T88806 CDOC86 303776 IC50 > 1000 nM T88806 C4U0BM 1878893 IC50 > 20000 nM T88806 C2E9ZX 3080994 IC50 = 1546000 nM T88806 C42AWQ 3797164 IC50 = 20500 nM T88806 CI51MD 9807891 IC50 > 500000 nM T88806 C68UYS 9808123 IC50 = 64 nM T88806 CK6A0I 9808598 IC50 > 500000 nM T88806 CB8GP1 9828375 IC50 = 26 nM T88806 CJ9HV0 9828819 IC50 = 20 nM T88806 C1OP9I 9828979 EC50 > 100000 nM T88806 C87ADQ 9830626 IC50 = 421 nM T88806 C13KPA 9848051 Ki < 10000 nM T88806 C04PAT 9849697 IC50 > 500000 nM T88806 CTM7V0 9851337 IC50 = 316 nM T88806 C2XD7P 9851886 IC50 > 100000 nM T88806 CN1R0K 9852055 IC50 > 500000 nM T88806 CR38MP 9853559 IC50 = 2200 nM T88806 C6E3OL 9863046 IC50 > 100000 nM T88806 C2ZAK6 9870468 IC50 > 800000 nM T88806 CHC56Q 9870640 IC50 = 640 nM T88806 C5EJN9 9884317 IC50 > 20000 nM T88806 CV4T6H 9885053 IC50 = 7800 nM T88806 CME97S 9894966 IC50 = 930 nM T88806 C04INH 9895205 IC50 > 100000 nM T88806 CNX29T 9907082 IC50 = 70000 nM T88806 C9QN4D 9919094 IC50 = 1100000 nM T88806 CF4J2Z 9923982 IC50 = 15000 nM T88806 CUBV32 9924032 IC50 > 20000 nM T88806 CCPD70 9927009 IC50 = 180000 nM T88806 CDU79H 9957105 IC50 = 95 nM T88806 C2R7TW 10069591 IC50 > 500000 nM T88806 C71AIN 10077862 IC50 > 30000 nM T88806 CO8D9C 10196873 IC50 = 133 nM T88806 C7U5CM 10336795 IC50 = 8000 nM T88806 C0IA8K 10455265 IC50 > 450000 nM T88806 CTZC60 10461016 IC50 > 100000 nM T88806 CY1JM2 11024622 IC50 = 1300000 nM T88806 CZO3H7 11399588 IC50 = 3.7 nM T88806 CX9G5B 11534748 IC50 = 25 nM T88806 CFZ2O9 11613998 IC50 = 1.6 nM T88806 CD87UQ 11627754 IC50 = 286 nM T88806 CXA2U4 11671832 IC50 = 670 nM T88806 CWU71P 11699824 IC50 = 15 nM T88806 CGU84F 11721315 IC50 = 1.7 nM T88806 C2ONX6 11721442 IC50 = 6 nM T88806 CT4D1K 11799915 IC50 > 100000 nM T88806 CS24BW 11973730 IC50 > 10000 nM T88806 CZTJ02 12795460 EC50 = 1031 nM T88806 CW41XZ 16663331 IC50 > 10000 nM T88806 CDUC32 16665100 IC50 = 2.5 nM T88806 CTGC60 16678135 IC50 = 2.3 nM T88806 C4T7ZE 16724119 IC50 = 1500 nM T88806 CU8YQ3 16756502 IC50 = 1.1 nM T88806 C9LF8T 16756503 IC50 = 445 nM T88806 CJUK37 16756504 IC50 = 155 nM T88806 C0KW3V 16756505 IC50 = 3.5 nM T88806 C04JOX 16756621 IC50 = 0.54 nM T88806 C4CU7T 16756622 IC50 = 0.55 nM T88806 CFH96E 16756623 IC50 = 0.8 nM T88806 CXK79J 16756847 IC50 = 231 nM T88806 CB15RX 16756849 IC50 = 86 nM T88806 CM18ZN 16756955 IC50 = 1.4 nM T88806 CL38IU 16756956 IC50 = 0.9 nM T88806 CW5P8L 16756957 IC50 = 0.55 nM T88806 CX6AR9 23627460 IC50 = 2 nM T88806 CAVY89 23636144 IC50 > 10000 nM T88806 C1VUH4 23636254 IC50 > 10000 nM T88806 C6LR7V 23636255 IC50 > 10000 nM T88806 C5MSF6 23636502 IC50 > 10000 nM T88806 CYND24 23729562 IC50 > 20000 nM T88806 C96PUZ 23729563 IC50 > 20000 nM T88806 CZ17YE 23731146 IC50 = 3900 nM T88806 CHXT18 23731243 IC50 = 4300 nM T88806 CEA9Z8 23731244 IC50 = 1200 nM T88806 CNK5O6 23731245 IC50 > 20000 nM T88806 C6W9OS 23731246 IC50 = 20000 nM T88806 C79OBD 24864541 IC50 = 82 nM T88806 CR72IF 24864718 IC50 = 11 nM T88806 CFRX87 24864719 IC50 = 710 nM T88806 C9L0QD 24864721 IC50 < 1 nM T88806 CXH2G0 24864898 IC50 < 1 nM T88806 CF23RY 24865076 IC50 = 8 nM T88806 CO3I0M 24865264 IC50 = 69 nM T88806 CPD30N 24865443 IC50 = 480 nM T88806 C17IUE 24865620 IC50 = 8 nM T88806 C7TPO5 24865624 IC50 = 2 nM T88806 C5DVB6 24865625 IC50 = 3 nM T88806 C5DYT6 24865999 IC50 = 24 nM T88806 C5JB3F 24866187 IC50 = 220 nM T88806 C8G2FE 24866358 IC50 = 2 nM T88806 C6I1OF 24866515 IC50 < 1 nM T88806 CZ7QL8 24866516 IC50 = 90 nM T88806 CNCH18 24866519 IC50 = 3 nM T88806 CY6WR2 24872066 IC50 = 2.1 nM T88806 CUM4E3 24872070 IC50 = 2 nM T88806 CG09DH 24872646 IC50 = 1.6 nM T88806 CRS65Q 24873110 IC50 = 2.2 nM T88806 C0HZ7E 24873345 IC50 = 2.7 nM T88806 C28KAH 24873465 IC50 = 43 nM T88806 C1PB6T 25025343 IC50 = 12 nM T88806 CDA2B9 25025730 IC50 = 130 nM T88806 CD2L7Z 25025937 IC50 < 1 nM T88806 C43TCR 25183860 IC50 = 5 nM T88806 CR92LD 25184415 IC50 = 7 nM T88806 C3J7GQ 28510125 IC50 = 136 nM T88806 CLX6T9 28510811 IC50 > 1000 nM T88806 C2SLU4 44286634 IC50 = 3100000 nM T88806 C7B6FS 44286652 IC50 = 65000 nM T88806 C47DUX 44320508 IC50 = 1000000 nM T88806 CX46NY 44343237 IC50 = 6100 nM T88806 C08QPE 44350169 IC50 = 3000 nM T88806 CELV48 44350342 IC50 = 0.18 nM T88806 CP4R1A 44350344 IC50 = 230 nM T88806 C14OBS 44350379 IC50 = 2700 nM T88806 CDE56C 44350392 IC50 = 18 nM T88806 C0W9CT 44350404 IC50 = 1500 nM T88806 CEP6G1 44350415 IC50 = 0.39 nM T88806 CR83VC 44350419 IC50 = 670 nM T88806 CX3MK8 44350425 IC50 = 4700 nM T88806 C4U0XW 44350427 IC50 = 310 nM T88806 CJ47ZT 44350428 IC50 = 13 nM T88806 CX09AV 44350435 IC50 = 1800 nM T88806 CX28UF 44350441 IC50 = 170 nM T88806 C7J9NH 44350447 IC50 = 21 nM T88806 CH6UX8 44350448 IC50 = 14 nM T88806 C4C2PF 44350449 IC50 = 39 nM T88806 CP4TD3 44350450 IC50 = 1.4 nM T88806 CR51ID 44378699 IC50 = 6000 nM T88806 CAO29R 44378701 IC50 = 100 nM T88806 CWP41H 44378720 IC50 = 4300 nM T88806 C2U6ZA 44378747 IC50 = 2100 nM T88806 CT9H2B 44378748 IC50 = 4500 nM T88806 CNS75M 44378858 IC50 = 830 nM T88806 CENU52 44378961 IC50 = 4300 nM T88806 C3UQT1 44378995 IC50 = 1560 nM T88806 CHC7N5 44379066 IC50 = 1200 nM T88806 CVYB52 44393453 IC50 > 20000 nM T88806 CAD12L 44393517 IC50 > 1000 nM T88806 C6G7RF 44436701 IC50 > 1000000 nM T88806 CZ1L9O 44436703 IC50 > 1000000 nM T88806 C7CAJ3 44436705 IC50 > 1000000 nM T88806 CR6XE2 44436707 IC50 = 18 nM T88806 CYOC34 44436708 IC50 > 1000000 nM T88806 CSF3V2 44436709 IC50 > 1000000 nM T88806 C67VHW 44436710 IC50 > 1000000 nM T88806 CBW09N 44436711 IC50 > 1000000 nM T88806 CRNQ31 44436712 IC50 > 1000000 nM T88806 C1YMJ2 44436713 IC50 = 170 nM T88806 CF4UR2 44436714 IC50 > 1000000 nM T88806 C52DMG 44436715 IC50 > 1000000 nM T88806 CLU84X 44436716 IC50 = 35100 nM T88806 CRO80K 44436717 IC50 = 57 nM T88806 CVGW76 44549110 IC50 = 0.3 nM T88806 CWL7J1 44549224 IC50 = 0.7 nM T88806 CO8EM6 44550577 IC50 = 0.1 nM T88806 CX1C4T 44552445 IC50 = 151.6 nM T88806 CCFW92 44605870 IC50 = 220 nM T88806 CM9VI1 44626482 IC50 = 1300 nM T88806 CBO95I 44626483 IC50 > 100000 nM T88806 CS36GK 44627949 IC50 = 520 nM T88806 CX6LM3 44628051 IC50 = 24 nM T88806 CVTO84 44628052 IC50 = 4700 nM T88806 CJQ37N 44628053 IC50 > 100000 nM T88806 CV4P3J 44628054 IC50 > 100000 nM T88806 CTU9W0 44628055 IC50 > 100000 nM T88806 C89ZFA 46224777 IC50 = 0.92 nM T88806 C5X1NZ 46224858 IC50 = 0.9 nM T88806 CDG6B1 46224859 IC50 = 351 nM T88806 CKM2X1 46224860 IC50 = 70 nM T88806 CL39GY 46224861 IC50 = 234 nM T88806 C56PVC 46226894 IC50 = 1.6 nM T88806 CVXH79 46226896 IC50 = 1.6 nM T88806 CBKZ57 46226897 IC50 = 1.5 nM T88806 C30JXH 46226899 IC50 = 13 nM T88806 C2WHK1 46226900 IC50 = 46 nM T88806 C5H9YT 46226901 IC50 = 65 nM T88806 CV8W7P 46226902 IC50 = 887 nM T88806 C83EWD 46226903 IC50 = 79 nM T88806 CRVU54 46226904 IC50 = 87 nM T88806 CE85AX 46226905 IC50 = 6.1 nM T88806 CP7U9T 50907449 IC50 = 19 nM T88806 CK7ZI0 56838719 IC50 = 1050 nM T88806 CG2NY0 57819421 IC50 = 466 nM T88806 CEG3V7 59665282 IC50 = 5900 nM T88806 C5MA9U 59665328 IC50 < 41 nM T88806 CR71ZG 59665343 IC50 = 150 nM T88806 CJ84CU 59665347 IC50 = 83 nM T88806 CTP16I 59665394 IC50 = 76 nM T88806 C5DJB3 59665402 IC50 = 140 nM T88806 C60EVZ 59665407 IC50 = 3 nM T88806 C4UH8X 59665418 IC50 = 6 nM T88806 C5RDW1 59665480 IC50 < 1 nM T88806 CSRE10 59665495 IC50 = 49 nM T88806 C1C0UT 68898764 IC50 = 21 nM T88806 CN93KB 68898863 IC50 = 39 nM T88806 CD10PM 68899361 IC50 = 9 nM T88806 CBF0K8 68899684 IC50 = 1900 nM T88806 C9LB1Y 68900219 IC50 = 1 nM T88806 C74UPO 68900657 IC50 = 9 nM T88806 CD4N6F 68901257 IC50 = 180 nM T88806 CK8UT9 68901290 IC50 = 110 nM T88806 CF4BZ9 68901306 IC50 = 1 nM T88806 CI0AL7 69244056 IC50 = 4 nM T88806 C31IUF 69863577 IC50 = 2807 nM T88806 CPF6S0 70681588 IC50 = 890 nM T88806 CQ4G2O 70683715 IC50 = 5 nM T88806 CVCJ03 70687988 IC50 = 2200 nM T88806 CX73MA 70689988 IC50 = 130 nM T88806 C92FXR 70690012 IC50 = 150 nM T88806 CPA07E 70694227 IC50 = 360 nM T88806 C8NZ7A 70694228 IC50 = 1 nM T88806 CM2AD4 70696326 IC50 < 1 nM T88806 C48NIF 70696327 IC50 = 970 nM T88806 CGMR28 71450831 IC50 = 1200 nM T88806 C8EM7Y 71550913 IC50 = 126.5 nM T88806 CY1MD5 71574157 IC50 = 7.3 nM T88806 C02ZBI 71574158 IC50 = 111 nM T88806 C16JKI 71574159 IC50 = 7 nM T88806 CU95LC 71574160 IC50 = 94 nM T88806 COJ8Y4 71574161 IC50 = 8.7 nM T88806 C5SG9H 71574261 IC50 = 115 nM T88806 C3C9QK 71574262 IC50 = 92 nM T88806 CTZU49 71574263 IC50 = 11 nM T88806 C4HB7F 71574264 IC50 = 39 nM T88806 C3S9QJ 71574355 IC50 = 72 nM T88806 C8V4UB 71574356 IC50 = 5.5 nM T88806 CX0SQ1 71574452 IC50 = 8.7 nM T88806 C1QE0K 71716365 IC50 = 197 nM T88806 CFYM81 71720633 IC50 = 27 nM T88806 CA9K6E 72204688 IC50 = 19 nM T88806 CLC7R0 72204689 IC50 = 9800 nM T88806 CCW43J 72204873 IC50 = 2100 nM T88806 CQ6TF8 72204875 IC50 = 9800 nM T88806 CC49AN 72204878 IC50 > 100000 nM T88806 C0N3SX 72205060 IC50 = 170 nM T88806 CZ2P8U 73345565 IC50 = 6600 nM T88806 CQAE56 73345568 IC50 > 10000 nM T88806 CU1VZ5 73345570 IC50 = 6400 nM T88806 CPT7S8 73345576 IC50 > 10000 nM T88806 C4P3JC 73346588 IC50 = 3650 nM T88806 CZ6Y9R 73347081 IC50 = 4190 nM T88806 CZ35TD 73347085 IC50 = 440 nM T88806 CGM9F7 73347087 IC50 = 7720 nM T88806 C89ENA 73347090 IC50 = 6800 nM T88806 CN1A2D 73347092 IC50 = 5190 nM T88806 CO9L2V 73348591 IC50 = 6240 nM T88806 C43LWV 73348592 IC50 = 1810 nM T88806 CM37AE 73348593 IC50 = 7200 nM T88806 C5BQ6R 73349139 IC50 = 57 nM T88806 CQ5D7B 73350175 IC50 = 870 nM T88806 CJEH13 73350177 IC50 = 6800 nM T88806 C20AJB 73350179 IC50 = 10000 nM T88806 C19PJE 73350181 IC50 = 4790 nM T88806 C2F3YZ 73351673 IC50 = 9200 nM T88806 CJA25I 73351674 IC50 = 2300 nM T88806 C6NCQ1 73351675 IC50 = 440 nM T88806 C46ULG 73351676 IC50 = 10000 nM T88806 C8B6NV 73351677 IC50 = 5100 nM T88806 CIYV49 73351678 IC50 = 1500 nM T88806 C20FGN 73353141 IC50 = 8700 nM T88806 CP6AJ3 73353143 IC50 = 8500 nM T88806 CUPR57 73353147 IC50 = 1200 nM T88806 C83RAM 73353150 IC50 = 8200 nM T88806 CAJ27W 73354663 IC50 = 7720 nM T88806 CT4A5S 73354664 IC50 = 4700 nM T88806 C6XTP9 73354667 IC50 > 10000 nM T88806 CZ1BL4 73354668 IC50 = 1230 nM T88806 C4EJK0 73356213 IC50 = 980 nM T88806 CH8G5C 73356216 IC50 > 10000 nM T88806 CPG36Q 73356217 IC50 = 6000 nM T88806 CD1S3N 73356221 IC50 = 840 nM T88806 C5ALQ2 76285468 IC50 = 74 nM T88806 CI07FE 90645591 IC50 = 66000 nM T88806 C8N6OE 90654504 IC50 = 108 nM T88806 C8TWH9 90654505 IC50 > 10000 nM T88806 CDVB75 90654506 IC50 > 10000 nM T88806 C5HG9N 90654507 IC50 = 64.2 nM T88806 CLCN89 117977916 IC50 = 63 nM T88806 CJO3B6 117978172 IC50 > 10000 nM T88806 C7ANO1 118709464 IC50 = 0.39 nM T88806 CY1IS6 118718872 IC50 = 10000 nM T88806 CV7DK0 122181680 IC50 > 1000 nM T88806 CWY3V2 122181682 IC50 > 1000 nM T88806 CRG07Q 124155531 IC50 > 10000 nM T88806 C69XPN 124163720 IC50 > 10000 nM T88806 C4R3BT 124163838 IC50 = 3200 nM T88806 CS2QR4 124163840 IC50 = 3200 nM T88806 C93HFX 127025140 IC50 = 15 nM T88806 CEU4X3 127025441 IC50 = 26 nM T88806 CTX71B 127025442 IC50 = 1500 nM T88806 C21ACR 133633869 IC50 > 1000 nM T88806 CPU86F 135438774 IC50 > 20000 nM T88806 C3JVT0 136152923 IC50 > 20000 nM T88806 C85WBP 137634338 IC50 = 95.8 nM T88806 C4IX7Z 137649002 IC50 = 30.7 nM T88806 C6NVW5 137652892 IC50 = 101.3 nM T88806 C0X8ER 145949722 IC50 = 20 nM T88806 C2MO7K 145951845 IC50 = 13 nM T88806 CG80FB 145951878 IC50 = 48 nM T88806 C1P0NL 145952828 IC50 = 22 nM T88806 CJA7N9 145953608 IC50 = 41 nM T88806 CZ4SK6 145954275 IC50 = 18 nM T88806 CTA08K 145956036 IC50 = 76 nM T88806 CY5I1O 145956101 IC50 = 45 nM T88806 C8RAG3 145956154 IC50 = 36 nM T88806 CCB51L 145956802 IC50 = 40 nM T88806 CTS5R3 145959048 IC50 = 28 nM T88806 CQ4ET5 145959752 IC50 = 31 nM T88806 CO0W4J 145961652 IC50 = 22 nM T88806 C23HZY 145971531 IC50 = 22 nM T88806 C75GFR 154734316 IC50 = 158 nM T88806 CR9DN2 154734318 EC50 = 9.9 nM T88806 C8ZUJ5 154734319 IC50 = 41.5 nM T88806 C17RZG 155515221 IC50 = 547 nM T88806 CHT1J6 155515540 IC50 = 72.9 nM T88806 CQ5C4M 155516533 IC50 = 689 nM T88806 CQNC74 155517321 IC50 > 10000 nM T88806 CRIA18 155519034 IC50 > 10000 nM T88806 C3S2YZ 155519712 IC50 = 563 nM T88806 CZY8F6 155520344 IC50 = 325 nM T88806 C9HB1M 155526953 IC50 = 5669 nM T88806 C2GJ5V 155527654 IC50 = 835 nM T88806 CQ1G0D 155528127 IC50 = 419 nM T88806 C2GSD7 155528224 IC50 = 3660 nM T88806 CPIL79 155528977 IC50 = 2722 nM T88806 C58JIQ 155530986 IC50 = 1.92 nM T88806 CJZU81 155532583 IC50 = 9287 nM T88806 C9T6SE 155533508 IC50 = 983 nM T88806 CJ7O2X 155534687 IC50 > 1000 nM T88806 C6TCP5 155546837 IC50 = 409 nM T88806 C6D2SM 155550380 IC50 > 10000 nM T88806 CWF98D 155552156 IC50 > 1000 nM T88806 CC64PJ 155561080 IC50 = 8029 nM T88806 C80PGY 155563043 IC50 = 5944 nM T88806 CEF3T8 155563936 IC50 = 38.4 nM T88806 C0SZJ1 155564443 IC50 = 1110 nM T88806 C98UME 155566748 IC50 = 2161 nM T88806 CY8S2L 155569251 IC50 = 11.9 nM T88806 C9NH4F 155569254 IC50 = 154 nM T88806 CZ9D2V 90645090 EC50 = 12 nM T88806 CWA6N4 90645092 EC50 = 763 nM T88806 CA8W7Q 90645094 EC50 = 365 nM T88806 D01AXA 11764797 IC50 = 259000 nM T88806 D06LUT 44379110 IC50 = 3440 nM T88806 D07WDB 104802 IC50 = 830000 nM T88806 D0A0KS 9851104 IC50 = 34700 nM T88806 D0B4JU 15409414 IC50 = 740 nM T20251 D00FGR 3599 IC50 > 100000 nM T20251 D00JAU 3749 IC50 = 194984.46 nM T20251 D00JVR 2267 IC50 = 100 nM T20251 D00KHM 16362 IC50 = 3.02 nM T20251 D00PEH 135449332 IC50 = 630.96 nM T20251 D00SBN 4746 IC50 = 7762.47 nM T20251 D00STL 644241 IC50 = 125.89 nM T20251 D00UVA 11556711 IC50 = 92100 nM T20251 D00UYE 4058 IC50 = 323.59 nM T20251 D00YLW 3033818 IC50 = 6025.6 nM T20251 D01AXB 60835 IC50 = 10000 nM T20251 D01AZG 5073 IC50 = 148 nM T20251 D01FGR 3100 IC50 = 2570.4 nM T20251 D01KPV 3348 IC50 = 21379.62 nM T20251 D01UTL 2995 IC50 = 1380.38 nM T20251 D01ZII 2726 IC50 = 1470 nM T20251 D01ZSO 4235 IC50 = 79432.82 nM T20251 D02EYG 10096344 IC50 > 30000 nM T20251 D02KOF 3948 IC50 = 2398832.92 nM T20251 D02MLW 60753 IC50 = 20 nM T20251 D02YIZ 12560 IC50 = 39 nM T20251 D03CJL 3168 IC50 = 32.2 nM T20251 D03CQE 5379 IC50 = 128824.96 nM T20251 D03DAP 3356 IC50 = 3890.45 nM T20251 D03DIG 5284371 IC50 = 301995.17 nM T20251 D03FLC 3878 IC50 = 251188.64 nM T20251 D03HFG 5324346 IC50 = 3100 nM T20251 D03IGH 213039 IC50 = 100000 nM T20251 D03MIR 3157 IC50 = 588.84 nM T20251 D03NHW 4583 IC50 = 1412537.54 nM T20251 D03QWT 73303 IC50 = 5011872.34 nM T20251 D04AAN 4078 IC50 = 320 nM T20251 D04CRN 54841 IC50 = 2100 nM T20251 D04FVU 6337614 IC50 = 1995.26 nM T20251 D04JCN 47811 IC50 = 120.23 nM T20251 D04JEE 4946 IC50 = 2828 nM T20251 D04LVK 57379345 IC50 = 1250 nM T20251 D04MSM 2554 IC50 = 104712.85 nM T20251 D04OSE 4485 IC50 = 50118.72 nM T20251 D04XGT 31593 IC50 > 100000 nM T20251 D04XPW 446220 IC50 = 4.4 nM T20251 D05CPV 208898 IC50 = 3000 nM T20251 D05EAM 4735 IC50 = 18800 nM T20251 D05LYX 3488 IC50 = 74000 nM T20251 D05MQK 110635 IC50 = 79432.82 nM T20251 D05OFX 219078 IC50 = 50118723.36 nM T20251 D05PIZ 15130 IC50 = 2187.76 nM T20251 D05SBO 46220502 IC50 = 10900 nM T20251 D05XGO 11154555 IC50 = 20720 nM T20251 D06ABF 3957 IC50 = 169.82 nM T20251 D06BCB 443955 IC50 = 39 nM T20251 D06GKN 2099 IC50 = 3235.94 nM T20251 D06MAJ 65906 IC50 = 350 nM T20251 D06MQM 6437380 IC50 = 8100 nM T20251 D06PZN 119584 IC50 = 4800 nM T20251 D06ZUK 3696 IC50 = 3388.44 nM T20251 D07KSG 2733526 IC50 = 1584.89 nM T20251 D07MVK 37393 IC50 = 40 nM T20251 D08CDI 208908 IC50 = 630957.34 nM T20251 D08JZS 4992 IC50 = 1100 nM T20251 D08VXO 6834 IC50 = 891.25 nM T20251 D08YIN 1727 IC50 = 4400000 nM T20251 D09EGZ 2719 IC50 = 2500 nM T20251 D09GOS 2812 IC50 = 3019.95 nM T20251 D09HNR 3002190 IC50 = 40000 nM T20251 D09KTS 24821094 Ki = 1100 nM T20251 D09MWJ 2092 IC50 = 125892.54 nM T20251 D09OJQ 4095 IC50 = 9772.37 nM T20251 D09QUQ 92253 IC50 = 20892.96 nM T20251 D09SGV 25154714 IC50 = 29200 nM T20251 D0AO5H 5578 IC50 = 239883.29 nM T20251 D0AR3J 439501 IC50 = 5800 nM T20251 D0AV3G 3151 IC50 = 162 nM T20251 D0B3UJ 115237 IC50 = 1000 nM T20251 D0B5LF 448042 Ki = 79432.82 nM T20251 D0B7NG 2725 IC50 = 1100 nM T20251 D0BD8D 6917698 IC50 = 12 nM T20251 D0BP9C 193962 IC50 = 25118.86 nM T20251 D0BZ7W 443879 IC50 = 125.89 nM T20251 D0C3SW 53465279 IC50 > 30000 nM T20251 D0C9SY 135400189 IC50 = 79432.82 nM T20251 D0CL9S 159269 IC50 = 5011872.34 nM T20251 D0CS2F 3955 IC50 = 33 nM T20251 D0D1AL 3559 IC50 = 10 nM T20251 D0D7KC 5488548 IC50 = 63095734.45 nM T20251 D0D9FV 4601 IC50 = 851.14 nM T20251 D0DK8V 2678 IC50 = 30199.52 nM T20251 D0DV3O 3241 IC50 = 100000 nM T20251 D0E1WI 3345 IC50 = 1819.7 nM T20251 D0E4DW 1775 IC50 = 100000 nM T20251 D0E6XR 3062316 IC50 = 15848.93 nM T20251 D0E7PQ 5311 IC50 > 30000 nM T20251 D0F0YZ 4737 IC50 = 22800000 nM T20251 D0G9YH 2179 IC50 = 208.93 nM T20251 D0GQ7K 4046 IC50 = 2600 nM T20251 D0GV8J 135565082 IC50 > 100000 nM T20251 D0H0KB 5070 IC50 > 25000 nM T20251 D0H3HM 60795 Ki = 598 nM T20251 D0H7AV 4820 IC50 = 20417.38 nM T20251 D0H7KF 5002 IC50 = 5754.4 nM T20251 D0I0DL 3689 IC50 = 100 nM T20251 D0I1FQ 54671008 IC50 > 50000 nM T20251 D0J0BU 10275777 Ki = 1800 nM T20251 D0J2KV 4932 IC50 = 440 nM T20251 D0JL2K 72474 IC50 = 50000 nM T20251 D0K3QS 6442177 IC50 = 15848931.92 nM T20251 D0K6GZ 60464 IC50 = 21700 nM T20251 D0K7WK 4595 IC50 = 812.83 nM T20251 D0L0ZF 5663 IC50 = 1096.48 nM T20251 D0L4YD 154059 IC50 = 251.19 nM T20251 D0L5WM 2157 IC50 = 10000 nM T20251 D0L7VL 3926 IC50 = 15.85 nM T20251 D0M4YC 3114 IC50 = 91201.08 nM T20251 D0N3VR 71616 IC50 > 40000 nM T20251 D0NJ3V 4680 IC50 = 7244.36 nM T20251 D0NR6S 3002977 IC50 = 79432.82 nM T20251 D0NS6H 3152 IC50 = 1995.26 nM T20251 D0NW3X 71329 IC50 = 5 nM T20251 D0O1WX 2764 IC50 > 30000 nM T20251 D0O3FG 125017 IC50 = 251188.64 nM T20251 D0O3OS 104850 IC50 = 4800 nM T20251 D0O8GK 71496458 IC50 = 16200 nM T20251 D0OB1J 39186 IC50 = 17300 nM T20251 D0P9RF 5401 IC50 = 17782.79 nM T20251 D0Q5UQ 214348 IC50 = 3981071.71 nM T20251 D0Q9EV 11965427 IC50 > 20000 nM T20251 D0R0FE 2520 IC50 = 10 nM T20251 D0R0MW 5329102 IC50 = 500 nM T20251 D0R1JV 60854 IC50 = 120.23 nM T20251 D0R1RS 3715 IC50 = 301995.17 nM T20251 D0RM9Q 68778 IC50 = 851.14 nM T20251 D0S5CU 4499 IC50 = 23000 nM T20251 D0T6WN 6451164 IC50 = 500 nM T20251 D0T8GD 89594 IC50 = 245470.89 nM T20251 D0T8XB 44513473 IC50 > 500000 nM T20251 D0TR5X 3386 IC50 = 10 nM T20251 D0U0VU 5312125 IC50 = 7943.28 nM T20251 D0U1OE 5452 IC50 = 33.2 nM T20251 D0U2JP 4369359 IC50 = 501187.23 nM T20251 D0U2OO 2477 IC50 = 3981.07 nM T20251 D0U3SY 49806720 IC50 > 30000 nM T20251 D0U5FS 3396 IC50 = 2300 nM T20251 D0U5GB 92727 IC50 = 8511.38 nM T20251 D0U5SI 4913 IC50 = 138038.43 nM T20251 D0V4QS 135398745 IC50 = 181.97 nM T20251 D0V8HJ 11671467 IC50 > 1000 nM T20251 D0W8WB 2353 IC50 = 3100 nM T20251 D0W9LX 2585 IC50 = 350 nM T20251 D0WE3O 5288826 IC50 = 1000000 nM T20251 D0WO8W 4062 IC50 = 154881.66 nM T20251 D0WV3U 4893 IC50 = 1584.89 nM T20251 D0X0RI 4178 IC50 = 10000 nM T20251 D0X4RN 3676 IC50 = 263026.8 nM T20251 D0X5ZI 6918493 IC50 = 501187.23 nM T20251 D0Y4JJ 2351 IC50 = 33 nM T20251 D0Y4QG 5388906 IC50 = 0.2 ug.mL-1 T20251 D0Y5AM 444031 IC50 = 79.43 nM T20251 D0Y5DO 2771 IC50 = 3981.07 nM T20251 D0Y5UG 2160 IC50 = 3280 nM T20251 D0Y7RW 4763 IC50 = 3019951.72 nM T20251 D0Z1RV 135398737 IC50 = 191 nM T20251 D0Z1UA 71301 IC50 = 316.23 nM T20251 D0Z1ZM 84029 IC50 = 33113.11 nM T20251 D0Z7ZM 135398744 IC50 = 3300 nM T20251 D00AUX 25230266 IC50 > 20000 nM T20251 D00BUR 216327 IC50 > 1000 nM T20251 D00DRL 44137946 IC50 > 30000 nM T20251 D00FHR 9865515 IC50 > 30000 nM T20251 D00IFR 58423153 IC50 > 30000 nM T20251 D00NZL 11955855 IC50 = 28100 nM T20251 D00RYA 16750271 IC50 > 10000 nM T20251 D00SWQ 10429242 IC50 > 100000 nM T20251 D00WDY 53477157 IC50 = 1400 nM T20251 D00XKB 57406537 IC50 = 2800 nM T20251 D01HLO 58438464 IC50 = 6900 nM T20251 D01NUR 118169620 IC50 = 69000 nM T20251 D01QSO 16654980 IC50 > 30000 nM T20251 D01UBY 46208367 IC50 > 50000 nM T20251 D01UUD 9948102 IC50 = 1700 nM T20251 D01ZAQ 25227436 IC50 > 100000 nM T20251 D02AIN 122678117 IC50 > 33000 nM T20251 D02AYL 456199 IC50 > 30000 nM T20251 D02DTQ 24745335 Ki = 3467.37 nM T20251 D02QWY 24785538 IC50 > 10000 nM T20251 D02WFN 46207733 IC50 = 60000 nM T20251 D03GNI 2166 IC50 = 3900 nM T20251 D03ISJ 135564632 IC50 > 30000 nM T20251 D03KHO 52934180 IC50 = 141000 nM T20251 D03KKR 3547 Ki = 25118.86 nM T20251 D03QAO 25008769 IC50 = 233000 nM T20251 D03QHC 49856296 IC50 = 13400 nM T20251 D03QIE 47953 IC50 = 44668.36 nM T20251 D03RIO 24743758 IC50 = 460 nM T20251 D04COD 25101874 IC50 = 588 ug.mL-1 T20251 D04JZH 11659955 IC50 = 30000 nM T20251 D04LOR 51030730 IC50 = 1900 nM T20251 D04LSD 9818903 Ki = 400 nM T20251 D04OSA 46202416 IC50 = 4800 nM T20251 D04QKU 11438771 IC50 = 7100 nM T20251 D04WUA 219101 IC50 = 10000 nM T20251 D05EXN 58298316 IC50 = 33000 nM T20251 D05LPW 25022354 IC50 = 79600 nM T20251 D05LRD 59286554 IC50 > 30000 nM T20251 D05UYQ 15984937 IC50 = 15848.93 nM T20251 D06DMQ 59472121 IC50 = 3000 nM T20251 D06ENM 66553195 IC50 = 6200 nM T20251 D06EPO 11192346 IC50 = 20000 nM T20251 D06TQR 76287260 IC50 = 26800 nM T20251 D06WHY 16747683 IC50 = 3200 nM T20251 D07EHV 44814409 IC50 = 12000 nM T20251 D07HPJ 11476171 IC50 = 130 nM T20251 D07HZG 11516136 IC50 = 126000 nM T20251 D07LWK 9811357 IC50 = 10000 nM T20251 D08AAV 46893585 IC50 > 100000 nM T20251 D08AOZ 86582336 IC50 = 5500 nM T20251 D08HOM 46207586 IC50 = 1000 nM T20251 D08QGT 17755052 IC50 = 64000 nM T20251 D08UUL 46700756 IC50 = 20000 nM T20251 D09NAW 60195662 Ki > 15857 nM T20251 D09OTX 89741565 IC50 = 1800 nM T20251 D09RVI 23649154 IC50 = 794.33 nM T20251 D0A3CL 49801838 IC50 = 22000 nM T20251 D0A7ZK 56944144 IC50 = 6100 nM T20251 D0B3FV 6445533 IC50 = 10300 nM T20251 D0B5HF 44476893 IC50 > 100000 nM T20251 D0C9UF 155805 IC50 = 1 nM T20251 D0CE6C 135565042 IC50 = 6300 nM T20251 D0DH5X 44472635 IC50 > 30000 nM T20251 D0E0JO 117857370 EC50 > 33000 nM T20251 D0EQ9T 24771368 IC50 > 10000 nM T20251 D0EY0A 42636350 IC50 > 32000 nM T20251 D0F0JJ 11560787 IC50 = 1200 nM T20251 D0F6YM 3035000 IC50 = 20000 nM T20251 D0F7PZ 53316710 IC50 = 12000 nM T20251 D0FD6D 11751922 IC50 = 20000 nM T20251 D0G6QV 208952 IC50 = 34860 nM T20251 D0H9DA 54761306 IC50 = 166000 nM T20251 D0HS5V 11234052 IC50 = 18000 nM T20251 D0HZ2E 5311271 Ki = 1100 nM T20251 D0I2XM 3038500 IC50 = 220 nM T20251 D0I3LO 91933883 IC50 > 10000 nM T20251 D0I3TU 45268455 Ki > 39000 nM T20251 D0I4PW 60164925 IC50 > 30000 nM T20251 D0IZ8X 90111638 IC50 > 10000 nM T20251 D0JU5X 400769 IC50 > 200000 nM T20251 D0K4FP 44548240 IC50 > 33000 nM T20251 D0K4HW 135409468 IC50 = 4466.84 nM T20251 D0K9IF 71666749 IC50 > 30000 nM T20251 D0L9KH 44623998 IC50 > 30000 nM T20251 D0L9QM 59568713 IC50 = 22000 nM T20251 D0LI1C 44469321 IC50 = 30440 nM T20251 D0LQ3L 77108121 IC50 = 195000 nM T20251 D0M3XR 46209133 IC50 = 39000 nM T20251 D0M4TJ 44219292 IC50 > 30000 nM T20251 D0M7CB 9919680 IC50 = 65700 nM T20251 D0M8FD 4261 IC50 > 30000 nM T20251 D0M8OC 16061509 IC50 > 10000 nM T20251 D0M9RQ 11697697 IC50 = 10000 nM T20251 D0MR0B 54766013 IC50 = 31040 nM T20251 D0N6NM 71721648 IC50 > 10000 nM T20251 D0N8QK 24743471 Ki = 8830 nM T20251 D0NU8J 117947097 IC50 > 50000 nM T20251 D0O0BM 44156901 IC50 = 8500 nM T20251 D0O1IM 58298318 IC50 > 33000 nM T20251 D0O1ZI 25006684 IC50 > 100000 nM T20251 D0O8BS 16039797 IC50 > 100000 nM T20251 D0O9XN 11691484 IC50 = 13000 nM T20251 D0OW9L 11973780 IC50 > 10000 nM T20251 D0P5CM 56945146 IC50 = 12589.25 nM T20251 D0PM5U 135564890 IC50 > 40000 nM T20251 D0PM7Q 11152667 IC50 = 15000 nM T20251 D0PW4N 6851740 IC50 = 4810 nM T20251 D0Q7RE 16007391 IC50 > 30000 nM T20251 D0QX8X 71479709 Ki = 3100 nM T20251 D0R0LB 91668194 IC50 > 100000 nM T20251 D0R2OU 25070031 IC50 = 13800 nM T20251 D0R3VK 42642654 IC50 = 4400 nM T20251 D0R8IU 24946280 IC50 > 100000 nM T20251 D0R9IU 44462758 IC50 = 8600 nM T20251 D0R9KG 11604525 IC50 = 11000 nM T20251 D0S1XX 134821691 IC50 > 80000 nM T20251 D0S5IR 86294073 IC50 > 30000 nM T20251 D0SG7B 49831257 IC50 = 85000 nM T20251 D0T0PN 9821217 Ki = 1800 nM T20251 D0T4QA 90456533 IC50 > 10000 nM T20251 D0U4FF 10437018 IC50 = 4000 nM T20251 D0U7KH 86567195 IC50 > 30000 nM T20251 D0U8QH 59239165 IC50 > 100000 nM T20251 D0V2YJ 11655511 IC50 = 20500 nM T20251 D0VI4N 90409366 IC50 > 10000 nM T20251 D0W8XT 60663 Ki = 190 nM T20251 D0XD4I 118502708 IC50 > 33000 nM T20251 D0XT0W 66555680 IC50 = 6900 nM T20251 D0XT6W 6918638 IC50 > 30000 nM T20251 D0Y3ZP 23480 IC50 = 500 nM T20251 D0Y5NA 118435360 IC50 = 9900 nM T20251 D0Y7NA 49871007 IC50 = 4500 nM T20251 D0Z2UQ 25262792 IC50 = 47500 nM T20251 D08IMD 16755780 IC50 = 23000 nM T20251 D0E2FZ 10149311 IC50 > 30000 nM T20251 D0HM5J 118253852 IC50 > 33000 nM T20251 D0IY0R 11591505 IC50 = 23600 nM T20251 D0X5OV 42609962 IC50 > 30000 nM T20251 D01KIJ 72545600 IC50 >= 18500 nM T20251 D02NRD 9865421 IC50 > 10000 nM T20251 D03GTM 118485599 IC50 = 69 nM T20251 D04MAZ 71731606 IC50 = 100000 nM T20251 D0AF0O 54670056 IC50 = 590 nM T20251 D0CV8T 874670 IC50 > 10000 nM T20251 D0D3GL 137662068 IC50 = 15000 nM T20251 D0D4OW 57338826 Ki > 100000 nM T20251 D0F8KE 71059525 Ki = 41.3 nM T20251 D0HG2S 86294663 IC50 = 67000 nM T20251 D0J1LK 118485649 IC50 = 490 nM T20251 D0LU9X 74221950 IC50 = 19000 nM T20251 D0NG8Q 75203906 IC50 = 20900 nM T20251 D0PJ8X 71562840 IC50 = 61700 nM T20251 D0PO8N 117881270 IC50 > 33000 nM T20251 D0V8FC 60169096 IC50 = 25000 nM T20251 D0WS3T 72706254 IC50 = 2700 nM T20251 D0YN2T 86302836 IC50 > 10000 nM T20251 D00PDG 44454750 IC50 = 800 nM T20251 D00PXQ 60785 Ki = 200 nM T20251 D02NGR 9934294 IC50 = 670 nM T20251 D03KWN 11373432 IC50 > 100000 nM T20251 D03OFO 9851380 IC50 = 6000 nM T20251 D04BQR 4342 IC50 = 100000 nM T20251 D06BPG 4528 IC50 > 27000 nM T20251 D06TGE 11226090 IC50 = 14200 nM T20251 D06VXY 9845214 IC50 = 420 nM T20251 D07BUO 25067561 IC50 = 19000 nM T20251 D07GIB 11614352 IC50 = 11000 nM T20251 D07KIJ 10008367 IC50 = 13000 nM T20251 D08AWI 11430856 Ki > 2000 nM T20251 D08SOF 5405 IC50 = 22 nM T20251 D09EVZ 507806 IC50 > 80000 nM T20251 D09RGW 11753159 IC50 > 15848.93 nM T20251 D09XHI 9879103 IC50 = 6350 nM T20251 D0A1NU 16049769 Ki > 45100 nM T20251 D0AQ3H 11505444 IC50 > 10000 nM T20251 D0B4TT 17747460 IC50 = 50.12 nM T20251 D0B7SP 11292933 Ki = 12589.25 nM T20251 D0E2PX 3087190 IC50 = 18.1 nM T20251 D0E3SD 9838729 IC50 > 33000 nM T20251 D0E6OA 65941 IC50 = 251.19 nM T20251 D0G1RH 6918446 IC50 = 194 nM T20251 D0H9GQ 9795276 IC50 = 10000 nM T20251 D0I5UU 123618 IC50 = 27.54 nM T20251 D0J0AE 10052040 IC50 > 3000 nM T20251 D0J9UI 9807238 Ki > 10000 nM T20251 D0K1VK 25262965 IC50 = 30400 nM T20251 D0N8NK 11641563 IC50 = 40000 nM T20251 D0OS6O 60149 IC50 ~ 3 nM T20251 D0Q3ES 11705608 IC50 = 3000 nM T20251 D0W7IR 9887884 IC50 = 32000 nM T20251 D0Y2HR 2247 IC50 = 0.9 nM T20251 D0Y6SN 5311096 IC50 = 630.96 nM T20251 D0Z0CH 3033962 IC50 = 5 nM T20251 C9H6CG 1287 IC50 = 6025.6 nM T20251 CXUC05 2215 IC50 = 2398.83 nM T20251 CCNZ53 2340 IC50 = 3981071.71 nM T20251 CPJ0C2 2747 IC50 = 8800 nM T20251 CZUI83 2769 IC50 = 6.457 nM T20251 CCW9O8 2825 IC50 = 1202.26 nM T20251 CYO1K2 2826 IC50 = 7244.36 nM T20251 C2AXN5 3148 IC50 = 12022.64 nM T20251 CDR20M 3185 IC50 = 1.2 nM T20251 C0H8GR 3191 IC50 = 331.13 nM T20251 C2XP5J 3255 IC50 = 72443.6 nM T20251 CY4WG9 3793 IC50 > 40000 nM T20251 C9LCD8 3823 IC50 = 1905.46 nM T20251 CP4RM6 4486 IC50 = 10000 nM T20251 C5ZC4S 5977 IC50 = 4365158.32 nM T20251 CP1QC0 9801 IC50 = 65 nM T20251 CBHG51 9822 IC50 > 10000 nM T20251 CZXE86 15330 IC50 = 2754.23 nM T20251 CN0WP7 15630 IC50 < 10000 nM T20251 CKCT41 28292 IC50 = 50118.72 nM T20251 CA12TG 38911 IC50 > 40000 nM T20251 C6GN7M 40692 Ki = 1900 nM T20251 CI93MP 51106 IC50 = 9100 nM T20251 C8ODZ3 56069 IC50 > 25000 nM T20251 CV4S2E 62969 IC50 = 200 nM T20251 CP8F7B 64143 IC50 = 12589.25 nM T20251 CD9TC8 64737 IC50 = 22000 nM T20251 C92TML 65014 IC50 > 100000 nM T20251 C97NOS 68634 IC50 = 2100 nM T20251 C1O4FS 73400 IC50 = 16000 nM T20251 CU1H3J 83952 IC50 = 316227.77 nM T20251 C7SXL6 87152 IC50 > 25000 nM T20251 C36LYP 104904 IC50 = 416869.38 nM T20251 C09TNA 107927 IC50 = 40000 nM T20251 CL4IR8 115159 IC50 = 50118.72 nM T20251 CR91WU 117964 IC50 = 84000 nM T20251 CZ48UK 117965 IC50 = 13000 nM T20251 CJ1XF0 119478 IC50 = 169824.37 nM T20251 CEP43C 122068 IC50 = 9500 nM T20251 C6SRK5 123942 IC50 = 1047.13 nM T20251 CMN95P 127718 IC50 = 20.89 nM T20251 CM01FR 128820 IC50 = 44000 nM T20251 CU0C6S 131698 IC50 = 491.4 nM T20251 CIG7L1 160023 IC50 = 8 nM T20251 CGSA42 163906 IC50 = 6100 nM T20251 CDB9P5 170922 IC50 < 10000 nM T20251 C7AV9Z 175533 Ki = 0.4 nM T20251 CLY60V 187063 IC50 = 6606.93 nM T20251 C97DNP 194450 IC50 = 4.3 nM T20251 CI2WO8 219099 IC50 = 120.23 nM T20251 C2V5FA 398712 IC50 = 5000 nM T20251 CLD6J9 441074 IC50 = 323.59 nM T20251 C1Z4HP 441362 IC50 = 5623.41 nM T20251 CQ0XH2 467825 IC50 = 10370 nM T20251 CKC8U4 507751 IC50 > 80000 nM T20251 CPXL01 507783 IC50 > 80000 nM T20251 CM40AT 507791 IC50 > 80000 nM T20251 CFY12E 516173 Ki > 10000 nM T20251 CNCR59 516203 Ki = 30000 nM T20251 C9MVL1 516212 Ki = 16000 nM T20251 CJUT37 516217 Ki = 5700 nM T20251 CRG4W0 516223 Ki = 3800 nM T20251 C2WHI5 516226 Ki = 22000 nM T20251 C9UOI0 516233 Ki = 8100 nM T20251 C67BKT 516235 Ki = 3000 nM T20251 CWTN29 516239 Ki > 10000 nM T20251 C6L1BX 516246 Ki = 3400 nM T20251 C4MQR0 516247 Ki = 5600 nM T20251 C1LB4X 516254 Ki = 37000 nM T20251 CQ52IA 516260 Ki = 14000 nM T20251 C65AZI 516264 Ki = 1000 nM T20251 COA04U 516275 Ki = 3500 nM T20251 C59YWP 516276 Ki = 9600 nM T20251 C9XU6R 516280 Ki = 6000 nM T20251 CHN28A 516284 Ki = 11000 nM T20251 CBYO78 516292 Ki = 2100 nM T20251 C4XN2D 516293 Ki = 2300 nM T20251 CUAO78 516314 Ki = 400 nM T20251 CF2J7U 592280 IC50 = 169824.37 nM T20251 C4TY8B 607867 IC50 = 74 nM T20251 C8WX7B 621620 IC50 = 109647.82 nM T20251 C2M9UC 656771 IC50 = 20 nM T20251 CP7U6Y 667468 IC50 = 6456.54 nM T20251 CN5CJ7 688803 IC50 = 99300 nM T20251 CZN6S9 743974 IC50 > 50118.72 nM T20251 CSMB29 759456 IC50 = 12400 nM T20251 C3LM4S 821286 IC50 > 100000 nM T20251 C90NZF 853261 IC50 > 10000 nM T20251 C79YAJ 1034176 IC50 = 1350 nM T20251 CT2VP9 1471775 IC50 > 32000 nM T20251 CK0JI9 1548955 IC50 = 181.97 nM T20251 C8JLO0 2243267 IC50 = 6300 nM T20251 CTZ4R5 2730286 IC50 = 1500 nM T20251 CD28JA 2735964 IC50 = 10000 nM T20251 CHTM19 2747356 Ki = 1538 nM T20251 C2J9ML 2781852 IC50 > 10000 nM T20251 CORX94 2804997 IC50 > 26302.68 nM T20251 CMRX81 2811640 IC50 > 10000 nM T20251 C9LDS2 2971413 Ki = 5418 nM T20251 C0F4YK 2980278 Ki > 40000 nM T20251 C14NBG 3008866 IC50 > 80000 nM T20251 CUY7J9 3008902 IC50 = 550 nM T20251 CE3Q4V 3008904 IC50 = 1300 nM T20251 CZ1V8Q 3008913 IC50 = 670 nM T20251 C1IS9G 3008917 IC50 = 150 nM T20251 CZV0O6 3008927 IC50 = 570 nM T20251 C8KY7B 3008930 IC50 = 1200 nM T20251 CSED31 3011729 IC50 = 13000 nM T20251 C3U7EZ 3035784 IC50 = 100 nM T20251 C2YQ0B 3082684 IC50 = 14000 nM T20251 CS5F1I 3083481 Ki = 1200 nM T20251 C3HJK8 3525815 IC50 = 2500 nM T20251 C8KN4J 3876755 IC50 > 10000 nM T20251 CO23EI 3959338 IC50 = 27300 nM T20251 C0TV9U 4227718 IC50 > 10000 nM T20251 C9INQ8 4390854 IC50 > 33000 nM T20251 CWE45H 4497898 IC50 = 27000 nM T20251 CO2SY7 4630909 Ki = 870 nM T20251 CE1CP8 4663848 IC50 = 33113.11 nM T20251 C3JHM8 4687521 IC50 = 100000 nM T20251 C16EGI 4961254 IC50 > 10000 nM T20251 CJP1K5 4987129 IC50 > 14790 nM T20251 CZ32RC 5230270 IC50 = 1445.44 nM T20251 CLNI10 5281408 IC50 = 773000 nM T20251 CJB7T6 5288494 IC50 > 33000 nM T20251 CW38FP 5311047 IC50 < 1000 nM T20251 C8EG4K 5326625 IC50 = 8100 nM T20251 C1OZS6 5436342 IC50 > 100000 nM T20251 C3Q2XB 5495793 IC50 > 80000 nM T20251 C0ZAM9 5495818 IC50 > 80000 nM T20251 C6SON9 5837004 IC50 = 36307.81 nM T20251 C95DOH 6098167 IC50 = 12000 nM T20251 CPV72R 6102824 IC50 = 3500 nM T20251 CGL87W 6483572 IC50 = 10500 nM T20251 CO9NP6 6890860 IC50 = 43620 nM T20251 CFTO93 6918704 IC50 = 710 nM T20251 CU68IK 7141881 IC50 > 10000 nM T20251 CZAN92 7472794 IC50 > 25000 nM T20251 C5J8HN 8902499 IC50 = 12700 nM T20251 CL9O2G 9390285 IC50 = 30000 nM T20251 C9IFX8 9390560 IC50 = 13000 nM T20251 CJ07ZA 9800555 IC50 = 32000 nM T20251 C5Z2KM 9805944 IC50 = 245 nM T20251 C2H4ZK 9806118 IC50 = 24 nM T20251 C1W2VB 9814248 IC50 = 5230 nM T20251 CAD92E 9815159 IC50 = 900 nM T20251 CTR6H5 9817349 IC50 = 1995.26 nM T20251 CJS5L9 9819317 IC50 > 30000 nM T20251 C71XRT 9821510 IC50 = 7199.99 nM T20251 CE6NF9 9823363 IC50 = 3100 nM T20251 CEL3C9 9824630 IC50 = 480 nM T20251 C0PQT8 9824969 IC50 = 39800 nM T20251 CZV60D 9825288 Ki = 26400 nM T20251 C97VAE 9825776 Ki = 22700 nM T20251 C8EC9B 9828617 IC50 = 2511.89 nM T20251 CWM26G 9830364 IC50 = 25118.86 nM T20251 C1FQ5A 9835490 IC50 = 8290 nM T20251 C0E7YV 9836903 IC50 > 30000 nM T20251 CU0HE4 9839392 Ki = 18 nM T20251 C30IAQ 9840150 IC50 = 5300 nM T20251 CXE1Y8 9842436 IC50 = 3200 nM T20251 CG3U7J 9843049 IC50 = 1100 nM T20251 CA6N0H 9843867 IC50 = 4700 nM T20251 C7VSU2 9845018 IC50 = 440 nM T20251 CT4E5Z 9846543 IC50 = 210 nM T20251 CKD2H4 9848990 IC50 = 7585.78 nM T20251 C9XY6D 9849838 Ki = 1180 nM T20251 CH57DZ 9850318 IC50 = 1413 nM T20251 CF72XZ 9860561 IC50 = 1600 nM T20251 CRBW42 9861124 IC50 = 5570 nM T20251 C3EX7S 9862272 IC50 = 204 nM T20251 CGC0F7 9864462 IC50 = 2760 nM T20251 CXZ6Q7 9866918 IC50 = 8200 nM T20251 CAOK24 9867098 IC50 = 80 nM T20251 CN9YD5 9868131 IC50 = 3000 nM T20251 C7T3VS 9870145 IC50 = 70 nM T20251 CK7FJ6 9870185 IC50 = 6309.57 nM T20251 CR0EG2 9879772 IC50 = 692 nM T20251 CQJ5X2 9879974 IC50 = 1240 nM T20251 CPS24V 9880847 IC50 = 27460 nM T20251 CS6FN7 9883254 IC50 > 100000 nM T20251 C9IR5L 9884379 IC50 = 90 nM T20251 C2TV9M 9884543 IC50 = 1100 nM T20251 CZ8C7G 9885279 Ki = 6800 nM T20251 C64EOU 9885465 Ki = 1000 nM T20251 CO84WK 9885754 Ki = 62000 nM T20251 C9I8ZU 9887120 IC50 = 10000 nM T20251 CUF35J 9887834 IC50 = 12600 nM T20251 C85BQG 9890458 IC50 = 14000 nM T20251 C2P3GS 9899500 IC50 = 2500 nM T20251 CE28TW 9900179 IC50 = 3020 nM T20251 C2Z9BL 9908431 Ki = 560 nM T20251 CYZ5N4 9909089 EC50 = 7.943 nM T20251 CHB5G9 9909904 IC50 = 199.53 nM T20251 CVJ7I8 9910573 IC50 = 176 nM T20251 C4B2QY 9913339 IC50 = 25000 nM T20251 CF4VO1 9914506 IC50 = 25118.86 nM T20251 CIW81R 9923839 IC50 = 3400 nM T20251 CQF2X8 9925089 IC50 = 974 nM T20251 C10VOI 9930235 IC50 = 3600 nM T20251 CANK40 9931593 IC50 = 10000 nM T20251 C1F4WB 9932192 IC50 = 6960 nM T20251 C9FZO7 9932679 IC50 = 10499.99 nM T20251 C5HQM7 9932974 IC50 = 150 nM T20251 C6RF9U 9933928 IC50 = 1000 nM T20251 CDY39E 9934161 IC50 > 5000 nM T20251 COP96L 9936388 IC50 = 1600 nM T20251 CV5X7E 9938284 Ki = 1000 nM T20251 CS58EO 9944019 IC50 = 3850 nM T20251 CX3ZK9 9946374 IC50 = 1190 nM T20251 CZ4X5D 9946965 IC50 = 101 nM T20251 CV1T2W 9947009 IC50 = 1620 nM T20251 CH6IJ8 9947172 IC50 = 1120 nM T20251 C8T1HO 9948670 Ki = 1300 nM T20251 CLR78W 9952894 Ki = 35000 nM T20251 CKF9X1 9953268 Ki = 1300 nM T20251 CMI58L 9956563 IC50 = 1.7 nM T20251 CJ6BV9 9959777 IC50 = 36 nM T20251 C1NPJ7 9965169 IC50 = 7390 nM T20251 CT7BR0 9965311 IC50 > 1000 nM T20251 C3KTF6 9965610 IC50 = 4670 nM T20251 C6CXJ3 9966330 IC50 = 4560 nM T20251 C0ORJ4 9966331 IC50 = 1310 nM T20251 C49MPX 9966437 IC50 = 3390 nM T20251 CJ2DK6 9966438 IC50 = 1480 nM T20251 C7ZK5J 9966516 IC50 > 10000 nM T20251 CC35UV 9966603 IC50 = 6830 nM T20251 CPX92V 9979309 Ki = 794.33 nM T20251 C7TPF5 9983233 Ki = 445 nM T20251 CGO70N 9983801 IC50 = 82 nM T20251 CJOV70 9983904 IC50 = 54000 nM T20251 CGEJ24 9985625 IC50 = 5100 nM T20251 CRYX90 9986337 IC50 = 9000 nM T20251 C7OAK1 9986346 IC50 = 25.12 nM T20251 CD86AJ 10000396 Ki = 85000 nM T20251 CUQF40 10003657 IC50 = 6309.57 nM T20251 CQL12P 10004545 IC50 > 5000 nM T20251 CGY63T 10004877 IC50 = 85000 nM T20251 CZW1M7 10005242 IC50 > 31622.78 nM T20251 C4Y8TH 10006938 IC50 = 14000 nM T20251 CE7IB5 10007642 IC50 = 11000 nM T20251 CCO68X 10008352 IC50 = 100 nM T20251 CUN7T8 10019811 Ki = 10000 nM T20251 C3NPS8 10025899 Ki = 1750 nM T20251 CA06TQ 10028888 IC50 = 6600 nM T20251 CI3Q9B 10030247 IC50 = 130 nM T20251 CWD3B7 10030344 IC50 = 400 nM T20251 C6V8MF 10032207 IC50 = 8300 nM T20251 C1WH8Q 10042344 IC50 > 10000 nM T20251 C90AVX 10044868 Ki = 51000 nM T20251 C04HZE 10046270 IC50 > 10 nM T20251 CA42DO 10047196 IC50 = 3000 nM T20251 C02OIU 10047339 IC50 = 2250 nM T20251 C73QBA 10047509 IC50 > 10 nM T20251 CR6NW9 10054055 IC50 = 5400 nM T20251 CH5SZ3 10073306 IC50 = 70000 nM T20251 CF7OC8 10073954 IC50 = 21000 nM T20251 CRQL64 10075375 Ki = 120 nM T20251 CR01QE 10076802 IC50 = 1800 nM T20251 C2BG6C 10085660 IC50 > 10000 nM T20251 C8G1PU 10087576 Ki = 2900 nM T20251 CH14BN 10089061 Ki = 480 nM T20251 CR17PA 10093856 IC50 = 2200 nM T20251 CS5K6Q 10095195 IC50 = 2000 nM T20251 C83ZDL 10096130 Ki = 2800 nM T20251 CTN9C2 10097082 IC50 = 3000 nM T20251 C9D5FP 10099787 Ki = 730 nM T20251 C3L9IN 10110435 IC50 = 34000 nM T20251 CBUX03 10113183 IC50 = 8950 nM T20251 CFY9M8 10115569 IC50 = 23000 nM T20251 CVK61T 10116047 IC50 = 26000 nM T20251 CD9EV1 10126599 Ki = 3600 nM T20251 C1WYS8 10127169 Ki = 46 nM T20251 C6N2TK 10131545 IC50 = 2150 nM T20251 CVZ3S9 10132138 IC50 = 10100 nM T20251 C26HWK 10132572 IC50 = 1310 nM T20251 CV67NU 10136016 IC50 = 16700 nM T20251 C09XVI 10144709 IC50 = 54 nM T20251 CLBD08 10144909 Ki = 850 nM T20251 CQM6E2 10149720 Ki = 20000 nM T20251 CLW3J6 10151756 IC50 = 5011.87 nM T20251 CB6V1X 10162604 Ki = 58400 nM T20251 C7JP1A 10163439 Ki = 610 nM T20251 C75JIV 10167216 Ki = 38100 nM T20251 CSHY89 10172243 Ki = 39000 nM T20251 CQ6JH8 10173083 Ki = 15000 nM T20251 CR80BV 10175126 IC50 > 30000 nM T20251 CW0OK6 10178465 IC50 = 6100 nM T20251 C85DYP 10183035 IC50 = 13600 nM T20251 C5K2GS 10185181 Ki = 200 nM T20251 C3DM7B 10186910 IC50 = 12200 nM T20251 CW98JD 10187118 IC50 = 400 nM T20251 C73LXY 10188021 Ki = 11 nM T20251 CK7UT9 10188786 Ki = 290 nM T20251 CLJ02H 10194468 Ki = 240 nM T20251 COV97M 10199905 IC50 = 18600 nM T20251 CCE6H8 10203632 IC50 = 36600 nM T20251 CO51ZR 10205659 Ki = 420 nM T20251 CISE26 10206059 IC50 = 89400 nM T20251 C51SKM 10209082 Ki = 25 nM T20251 CK72XG 10209108 Ki = 490 nM T20251 CCG65P 10210026 Ki = 1200 nM T20251 CT2N1Z 10222208 Ki = 840 nM T20251 C18FMW 10237542 Ki = 320 nM T20251 CQGN38 10237827 Ki = 29 nM T20251 C2PLB1 10239891 IC50 > 30000 nM T20251 C8PJ1V 10248119 IC50 > 10000 nM T20251 CZ90LD 10250452 IC50 = 4600 nM T20251 C24QZK 10256734 IC50 = 4000 nM T20251 CXJ2O5 10256826 IC50 = 2000 nM T20251 C3OE5Z 10257392 IC50 = 2100 nM T20251 C67GCK 10258336 Ki = 43 nM T20251 CF2M9O 10268223 IC50 = 234 nM T20251 CGRQ23 10274114 IC50 = 2700 nM T20251 CHY71P 10274246 IC50 = 960 nM T20251 CM6SE7 10280445 IC50 = 4400 nM T20251 CMNH04 10286136 IC50 = 3300 nM T20251 CUQC81 10287415 Ki = 9400 nM T20251 C9K0SA 10288761 IC50 = 5000 nM T20251 CT89LX 10297708 IC50 = 4000 nM T20251 CV10CU 10297977 Ki = 100 nM T20251 C90DYG 10297996 IC50 = 50100 nM T20251 C1AP6H 10298858 Ki = 2100 nM T20251 CAX9W2 10302405 Ki = 34 nM T20251 C1W5ZD 10308681 Ki = 8050 nM T20251 C3M1VR 10309552 Ki = 225 nM T20251 CZ18PL 10316203 IC50 = 7500 nM T20251 C26EKI 10316979 IC50 = 31000 nM T20251 CF1S8U 10320144 IC50 = 86000 nM T20251 C03ZKG 10324551 IC50 = 5000 nM T20251 CBA2C6 10325032 IC50 = 224 nM T20251 CLKX29 10335984 Ki = 4500 nM T20251 CEZ95L 10342016 Ki = 52000 nM T20251 C5MH7Y 10343434 IC50 = 300 nM T20251 CW50TU 10345610 IC50 = 35200 nM T20251 CIYQ04 10358984 Ki = 6300 nM T20251 CGQN51 10359235 IC50 > 30000 nM T20251 CT6Y9I 10365686 IC50 = 38000 nM T20251 CFH29X 10367570 IC50 = 300 nM T20251 CDA5F7 10369999 IC50 = 6200 nM T20251 C2KO8V 10388264 IC50 = 29000 nM T20251 CP7CH6 10389946 IC50 = 38000 nM T20251 C3H9SB 10390717 IC50 = 19700 nM T20251 CJQV19 10391684 IC50 > 80000 nM T20251 CM9R2K 10391877 IC50 = 1200 nM T20251 CCZ17H 10392978 IC50 = 844 nM T20251 C9WC5D 10393066 IC50 > 8900 nM T20251 CU6X7E 10393880 IC50 = 130 nM T20251 C59QRY 10393962 Ki = 950 nM T20251 C76WZF 10401439 Ki = 11000 nM T20251 CG1T4B 10405623 IC50 = 2700 nM T20251 C6EJ8D 10410012 IC50 = 6.2 nM T20251 C56SLV 10412648 IC50 = 38 nM T20251 CV60SK 10413034 IC50 > 30000 nM T20251 CBN4H0 10415698 IC50 = 1300 nM T20251 CW80YU 10415870 Ki = 710 nM T20251 CUZE30 10416011 IC50 = 100 nM T20251 C6GXW2 10426299 Ki = 1200 nM T20251 C6KR8Z 10428027 Ki = 5100 nM T20251 CS7FG5 10429706 IC50 = 2570.4 nM T20251 C5ZXU8 10433753 IC50 = 25000 nM T20251 C5GQF1 10436125 IC50 = 22700 nM T20251 CWCA76 10439426 IC50 = 76000 nM T20251 C80TCL 10450279 Ki = 5000 nM T20251 CQ4C7Y 10450926 IC50 = 28600 nM T20251 CHW2U1 10451701 IC50 > 33000 nM T20251 C1T7QW 10456093 IC50 = 11000 nM T20251 CVSP85 10456367 IC50 = 29000 nM T20251 C8DWH6 10456892 IC50 = 30700 nM T20251 C38VGA 10457264 IC50 = 2000 nM T20251 C10NHR 10457710 IC50 = 2000 nM T20251 CMDU71 10460463 IC50 = 100 nM T20251 CWFK56 10461282 IC50 = 660 nM T20251 CGXY36 10482372 IC50 = 18100 nM T20251 CEW7C9 10482996 IC50 = 400 nM T20251 C7YPV6 10483558 IC50 = 250 nM T20251 CB52TQ 10495305 Ki = 3000 nM T20251 CPG8U3 10495787 Ki = 1500 nM T20251 C7W9LB 10498834 IC50 = 400 nM T20251 CI0PU7 10518508 IC50 = 10.96 nM T20251 CUQ03E 10520440 Ki = 1600 nM T20251 C2B9PT 10522146 Ki = 930 nM T20251 CV57XZ 10546579 Ki = 110 nM T20251 CMK39Q 10553487 IC50 > 10000 nM T20251 C8E1UH 10570940 IC50 = 3000 nM T20251 CKYT25 10597785 IC50 = 8800 nM T20251 C74NSJ 10615016 Ki = 7000 nM T20251 CQ75TL 10640054 Ki = 1400 nM T20251 C8C2GN 10640055 Ki = 2100 nM T20251 CY9A6G 10689687 IC50 = 790 nM T20251 CG0M4S 10697284 IC50 = 2400 nM T20251 COQ25N 10697363 IC50 = 100 nM T20251 C49IUL 10708935 Ki > 1100 nM T20251 C52SWI 10711404 Ki > 7000 nM T20251 C7PDA6 10713670 Ki = 500 nM T20251 C18ZBG 10758132 Ki = 238 nM T20251 CDK53W 10763704 IC50 = 1000 nM T20251 CFH1Q4 10805130 Ki = 2500 nM T20251 CDOH18 10851309 Ki = 8200 nM T20251 C0VQ3C 10853014 Ki = 5400 nM T20251 CV6ZN3 10861900 Ki = 710 nM T20251 C9QUV7 10863652 Ki = 25000 nM T20251 CX3RT7 10874250 IC50 = 180 nM T20251 C6KW8J 10884405 IC50 = 4300 nM T20251 C4QZ2E 10895064 IC50 = 5800 nM T20251 CLI84D 10895869 IC50 = 9900 nM T20251 C5L2FR 10896860 IC50 = 110 nM T20251 CZFJ03 10899797 IC50 > 60000 nM T20251 CAB0O8 10906012 IC50 = 2700 nM T20251 CDR7G5 10925892 Ki = 69 nM T20251 C9OI8S 10927262 Ki = 1900 nM T20251 CD10XK 10928028 IC50 = 4700 nM T20251 CR8NL2 10950878 IC50 = 870 nM T20251 C4PK7X 10971209 Ki = 570 nM T20251 C6HI0W 10971692 IC50 = 8399.99 nM T20251 C0BUR1 10991521 Ki = 110 nM T20251 CE6XI4 10993905 IC50 = 190 nM T20251 C3WI1P 11004853 IC50 = 4400 nM T20251 CH2A4Z 11016041 IC50 = 4900 nM T20251 C0A7DI 11017241 Ki = 39000 nM T20251 C1N5EF 11026589 IC50 = 9099.99 nM T20251 CG9JC8 11036563 Ki = 4000 nM T20251 C5P8RW 11048955 Ki = 22400 nM T20251 C0EWV4 11056631 Ki = 47 nM T20251 CEPM03 11068867 IC50 = 5870 nM T20251 C56YON 11069321 IC50 = 77 nM T20251 CKBM74 11070099 IC50 = 220 nM T20251 CG2WF1 11111531 Ki = 251 nM T20251 CHX96W 11133309 Ki = 7143 nM T20251 C0VBZ4 11144668 IC50 = 11999.99 nM T20251 CLU8C6 11145028 IC50 = 10000 nM T20251 C7HM0O 11152739 IC50 = 9200 nM T20251 C4NAJ5 11154544 IC50 = 1600 nM T20251 C76YFB 11155030 IC50 = 3300 nM T20251 C3X0AC 11155482 IC50 = 65000 nM T20251 C9AT4X 11163693 IC50 > 20000 nM T20251 CDY8S7 11165745 IC50 = 1650 nM T20251 CK67YW 11166256 Ki > 150000 nM T20251 C6FX8E 11166272 IC50 = 7700 nM T20251 C7OEX0 11174494 IC50 = 17200 nM T20251 CI7L1C 11176908 IC50 = 10000 nM T20251 C1QWM8 11178027 IC50 = 27000 nM T20251 CPEV03 11178961 IC50 = 466 nM T20251 C3TW2O 11187225 IC50 = 2700 nM T20251 C6EWJ9 11188910 IC50 = 13000 nM T20251 C3CAP9 11189372 IC50 = 1000 nM T20251 CUBX19 11189444 IC50 = 1300 nM T20251 CAN73X 11189693 IC50 = 730 nM T20251 CDOC09 11199458 IC50 = 33500 nM T20251 CE6HS7 11200189 IC50 = 56700 nM T20251 CC25EY 11200344 IC50 = 9900 nM T20251 CP6UL9 11200377 IC50 = 9800 nM T20251 CIAE47 11211122 IC50 = 44113 nM T20251 CS5ET8 11212373 IC50 = 1800 nM T20251 CY57AG 11212679 Ki = 794.33 nM T20251 CQ1E8L 11213136 IC50 = 1000 nM T20251 C20HPU 11220991 IC50 = 2300 nM T20251 C5TAN7 11223519 IC50 = 15000 nM T20251 C1VM2S 11225043 IC50 = 200 nM T20251 C0FSV9 11225074 IC50 = 1400 nM T20251 CP9Z1V 11225445 IC50 = 440 nM T20251 CHC3F8 11226573 IC50 = 820 nM T20251 CU75LJ 11227168 IC50 = 26000 nM T20251 CA39QR 11227406 IC50 = 400 nM T20251 C6D3UR 11237434 IC50 = 17900 nM T20251 CC62PB 11238080 IC50 = 52 nM T20251 CTS6F4 11238521 IC50 = 460 nM T20251 C8J5KI 11238580 IC50 = 750 nM T20251 CP8EW3 11245596 IC50 > 10000 nM T20251 C8TD3U 11247946 IC50 = 900 nM T20251 CX43IH 11248146 IC50 = 700 nM T20251 CW1O5V 11256620 IC50 = 220 nM T20251 CP0C2Q 11257803 IC50 > 11000 nM T20251 CZ98EU 11259253 IC50 = 3.6 nM T20251 C7XI0R 11260032 IC50 = 794.33 nM T20251 C92CYH 11265950 Ki > 3000 nM T20251 CRZ3V0 11269310 IC50 = 11784 nM T20251 C2U7OP 11270012 IC50 = 1800 nM T20251 C3N1MF 11270500 IC50 > 24000 nM T20251 C26HWL 11270869 IC50 = 560 nM T20251 CRDU42 11271947 IC50 = 12000 nM T20251 CL0DP6 11272440 IC50 = 501.19 nM T20251 CK36XS 11273324 IC50 = 83.18 nM T20251 CZ8DU0 11273379 IC50 = 10000 nM T20251 C53DQM 11273508 IC50 = 100 nM T20251 COV2U9 11281200 IC50 = 1700 nM T20251 C83KDF 11281738 Ki > 150000 nM T20251 C8CS5F 11282651 IC50 = 6900 nM T20251 CP27SY 11283686 IC50 = 1300 nM T20251 C9X0TH 11291017 IC50 = 15000 nM T20251 CNE3Z7 11296572 IC50 = 700 nM T20251 CV1LG4 11301893 IC50 = 1100 nM T20251 C9BLC7 11304596 Ki = 1995.26 nM T20251 CIMB79 11305766 IC50 = 199.53 nM T20251 C9L0IK 11313056 IC50 = 300000 nM T20251 C30MLR 11313946 IC50 > 31600 nM T20251 CNT19Q 11315446 IC50 = 11000 nM T20251 CVB45M 11315811 IC50 = 24000 nM T20251 C8S4FU 11317045 IC50 = 600 nM T20251 C5DBK1 11326750 IC50 > 50000 nM T20251 CWT28O 11328029 IC50 = 11.5 nM T20251 CP8Y7T 11328449 IC50 = 1800 nM T20251 C5M3ZN 11329138 IC50 = 6100 nM T20251 CQ1CG9 11330529 IC50 = 30000 nM T20251 CIT2Y7 11330837 IC50 > 30000 nM T20251 C7O0ER 11337925 IC50 = 5094 nM T20251 CKZ20A 11353843 IC50 = 9000 nM T20251 CX6C2M 11353855 IC50 = 28000 nM T20251 C0PUK5 11360073 IC50 = 20500 nM T20251 C9L7AT 11364901 IC50 = 40 nM T20251 CZ82WH 11365166 IC50 > 30000 nM T20251 C4BZ1C 11372427 IC50 = 20000 nM T20251 COH57K 11373894 Ki = 1000 nM T20251 C25ZCN 11374110 IC50 > 30000 nM T20251 C36OES 11374857 IC50 = 3.6 nM T20251 CWO2A7 11382160 IC50 = 62000 nM T20251 C2E8MJ 11382472 IC50 = 11989 nM T20251 CEKP86 11383454 IC50 = 501.19 nM T20251 CO1I8H 11384634 Ki = 885 nM T20251 CL1W3C 11387497 IC50 = 100 nM T20251 CE2M9F 11387511 IC50 = 13000 nM T20251 CCK08I 11388055 IC50 = 650 nM T20251 C53ANS 11393281 IC50 > 30000 nM T20251 C9AOM3 11397017 IC50 = 470 nM T20251 CF4OX6 11397149 Ki = 316.23 nM T20251 C7M3XJ 11397742 IC50 = 22600 nM T20251 C82ERW 11397777 IC50 = 350 nM T20251 CQE92F 11406708 IC50 = 21079 nM T20251 CE5ZK6 11409228 IC50 > 30000 nM T20251 CMW42X 11416123 IC50 > 20000 nM T20251 C6I0YP 11416924 IC50 = 3000 nM T20251 C6BE9Q 11417954 IC50 = 78000 nM T20251 CFX98O 11418182 Ki = 5561 nM T20251 C2N0AG 11421712 IC50 > 30000 nM T20251 CML2H3 11428837 IC50 = 7900 nM T20251 CREQ51 11429654 IC50 > 30000 nM T20251 C1YV6P 11442292 IC50 > 100000 nM T20251 CKU8Y3 11442383 IC50 = 18000 nM T20251 CG58SO 11444350 IC50 = 6309.57 nM T20251 CC9D4O 11444936 IC50 = 100 nM T20251 C07VBT 11445050 IC50 = 1900 nM T20251 CY7HT3 11452117 IC50 = 766 nM T20251 CQTM82 11452706 Ki > 150000 nM T20251 CE42DM 11453673 Ki = 1000 nM T20251 CP1WH5 11461365 Ki = 1100 nM T20251 CF6DQ2 11462727 IC50 = 40000 nM T20251 CKU5J7 11464405 IC50 = 4 nM T20251 C39QNY 11464915 IC50 = 500 nM T20251 CO95HP 11474838 IC50 = 19750 nM T20251 C3GMQ1 11477018 IC50 = 794.33 nM T20251 CH6X2L 11478011 IC50 = 6400 nM T20251 CRJ90F 11478858 IC50 = 870 nM T20251 C69PFD 11484605 IC50 > 30000 nM T20251 C8BY4A 11489501 IC50 = 501.19 nM T20251 CA8KE0 11492902 Ki > 20000 nM T20251 C1O9XD 11493620 IC50 = 240 nM T20251 CV41ER 11494867 IC50 = 2400 nM T20251 CXW96U 11495012 IC50 = 18000 nM T20251 CMQ86R 11495432 IC50 = 2530 nM T20251 C7H9AB 11495849 IC50 > 100000 nM T20251 CPX26I 11496746 IC50 = 50118.72 nM T20251 C5Z7GQ 11497411 IC50 = 251.19 nM T20251 CL17QT 11497455 IC50 > 10000 nM T20251 C9YU1O 11497679 IC50 = 1000 nM T20251 CQT5U8 11497680 IC50 = 1995.26 nM T20251 C9JD4N 11497924 IC50 = 1000 nM T20251 C69AMJ 11500781 IC50 = 910 nM T20251 C3B0LO 11501191 IC50 = 760 nM T20251 C6HM0U 11501983 IC50 > 10000 nM T20251 CZIE58 11502008 IC50 = 8.1 nM T20251 CI62OX 11502343 IC50 = 1800 nM T20251 CPO8S1 11502381 IC50 = 7900 nM T20251 CGB8M5 11502401 Ki = 30 nM T20251 C2TVA0 11502638 IC50 = 3800 nM T20251 C3ME1U 11502912 IC50 = 20000 nM T20251 C3ROH5 11504077 IC50 = 2511.89 nM T20251 COD9Z2 11504477 IC50 = 1300 nM T20251 CFSH67 11504490 IC50 = 10000 nM T20251 C10FVQ 11505089 IC50 = 800 nM T20251 C97WGN 11505187 IC50 = 7700 nM T20251 CHX56T 11508058 IC50 = 20200 nM T20251 CLPO39 11508317 Ki = 1100 nM T20251 CH75CA 11508844 IC50 = 4000 nM T20251 C7G4VM 11508924 IC50 = 12000 nM T20251 CV4IZ7 11509189 IC50 = 3036 nM T20251 CCP2Z0 11510399 IC50 = 1370 nM T20251 C72BCW 11510887 IC50 = 13.5 nM T20251 C1LCD7 11510932 IC50 = 560 nM T20251 CF45XR 11511026 Ki = 10 nM T20251 COT4H9 11511117 IC50 = 10000 nM T20251 CE62TB 11511267 IC50 = 1500 nM T20251 C2T8YD 11511361 IC50 > 10000 nM T20251 CP8B7T 11511719 IC50 > 10000 nM T20251 C9DE5V 11511776 IC50 = 490 nM T20251 CDQ18N 11515125 IC50 > 5000 nM T20251 CP9RB7 11515387 Ki > 3000 nM T20251 C23DKS 11516307 Ki = 160 nM T20251 CO0T6Q 11516310 Ki = 910 nM T20251 CS24AX 11516386 IC50 = 2800 nM T20251 CNM42D 11516387 IC50 = 5000 nM T20251 C6X1AJ 11516392 Ki = 710 nM T20251 CZ4OM7 11516508 IC50 = 1730 nM T20251 CVNP35 11517292 IC50 > 3200 nM T20251 C20FMG 11517340 IC50 = 10000 nM T20251 CPQN50 11517341 IC50 = 10000 nM T20251 CTA7M3 11517739 IC50 = 4600 nM T20251 CG3BZ9 11517980 IC50 = 137000 nM T20251 CW68BJ 11518143 IC50 = 14500 nM T20251 CLGO54 11518300 IC50 = 9190 nM T20251 C1KL7T 11518341 IC50 = 4000 nM T20251 CZ3D5Y 11518933 IC50 > 10000 nM T20251 C0WU7G 11518972 IC50 = 125.89 nM T20251 CM4B3J 11519133 IC50 = 6309.57 nM T20251 C08JSL 11519134 IC50 = 5011.87 nM T20251 CY47AQ 11519784 IC50 > 10000 nM T20251 C04RCG 11519858 IC50 = 7943.28 nM T20251 CM09RF 11524148 Ki = 690 nM T20251 CL09JW 11524225 IC50 = 2000 nM T20251 CBRO68 11524900 Ki = 4100 nM T20251 CU7B8I 11525190 IC50 = 110000 nM T20251 CR83WI 11525569 IC50 = 2500 nM T20251 CTNX29 11526451 IC50 = 1000 nM T20251 CR9NA7 11526531 IC50 = 1000 nM T20251 C0O3XD 11527019 IC50 = 58500 nM T20251 CEX8Y5 11527102 IC50 > 10000 nM T20251 CNL15V 11527195 IC50 = 10000 nM T20251 C0BF5R 11527661 IC50 > 30 nM T20251 C75FPD 11529874 Ki = 2840 nM T20251 C0BC6Y 11530223 Ki > 5000 nM T20251 C7NO5X 11531213 Ki = 1000 nM T20251 CZ93HX 11531536 Ki = 710 nM T20251 C94AGK 11531634 Ki = 5000 nM T20251 CS7Q6G 11532065 Ki = 70 nM T20251 CDX19H 11532153 Ki = 42 nM T20251 C89JTB 11532924 IC50 = 1800 nM T20251 C4W2IN 11533195 IC50 = 23900 nM T20251 CFU5V9 11533398 Ki = 800 nM T20251 CJF92G 11533429 IC50 = 3981.07 nM T20251 C2EQ1U 11533448 IC50 = 3981.07 nM T20251 C4LOQ9 11533473 IC50 = 1258.93 nM T20251 CZW9U3 11534726 IC50 = 1995.26 nM T20251 CR53ZL 11537871 IC50 = 18000 nM T20251 C29LCK 11537876 IC50 > 63000 nM T20251 C7R3HN 11538251 Ki = 2200 nM T20251 C8GZ1I 11539020 IC50 = 10000 nM T20251 CIR9M2 11539598 Ki = 16 nM T20251 CSN91H 11539722 IC50 = 6309.57 nM T20251 CJGL17 11539751 IC50 = 19054.61 nM T20251 C0J9NF 11539823 Ki = 3800 nM T20251 CIJ51X 11539903 IC50 = 38000 nM T20251 C0X6CJ 11540474 IC50 = 5011.87 nM T20251 CFS7T8 11540675 IC50 = 17100 nM T20251 CBR9K8 11541314 IC50 > 100000 nM T20251 C8P5GF 11541506 Ki > 10000 nM T20251 CY0JX9 11541985 IC50 = 8428 nM T20251 C5JEZ9 11544171 IC50 < 31622.78 nM T20251 C9UG2V 11544758 Ki > 40000 nM T20251 CS0B4G 11544795 IC50 = 940 nM T20251 CX0DJ3 11545423 Ki = 8252 nM T20251 CF52ZB 11545686 IC50 = 5940 nM T20251 CGE5W7 11546121 Ki = 2800 nM T20251 CFNG56 11546387 Ki = 430 nM T20251 CHT8D7 11547260 IC50 > 30000 nM T20251 CD14OF 11547466 IC50 = 1000 nM T20251 C61LDE 11548217 IC50 = 630.96 nM T20251 CKZ9B0 11548239 IC50 = 158.49 nM T20251 CPA7K8 11548755 IC50 = 251.19 nM T20251 C34JAV 11551351 Ki > 5000 nM T20251 C3DG8U 11552010 IC50 = 340 nM T20251 CCLR26 11552773 IC50 = 19000 nM T20251 CKGI84 11553070 IC50 = 2100 nM T20251 CH0E4A 11553554 Ki = 3100 nM T20251 CKT1O8 11554040 Ki = 2600 nM T20251 CA16WP 11554165 IC50 > 90000 nM T20251 CZD24Q 11554412 IC50 = 47400 nM T20251 CMC79Y 11554762 Ki = 4200 nM T20251 C0VMG7 11555265 IC50 = 251.19 nM T20251 C64NID 11555572 IC50 = 16000 nM T20251 C3Y4GR 11555971 IC50 = 5011.87 nM T20251 CNWU65 11556070 IC50 = 1750 nM T20251 C3RMI1 11559300 IC50 = 5030 nM T20251 C5WKO2 11559625 IC50 > 10 nM T20251 CXR53E 11561126 IC50 = 30 nM T20251 CX1VD8 11562113 IC50 = 1258.93 nM T20251 C0JU9T 11562199 IC50 = 5011.87 nM T20251 CD9SM0 11562361 IC50 > 10000 nM T20251 CQ8CJ9 11562662 IC50 = 10000 nM T20251 C7B4YX 11563243 Ki > 10000 nM T20251 C1VF0P 11566266 IC50 = 1080 nM T20251 CDP9Z0 11566316 IC50 > 20000 nM T20251 C8C1VW 11566318 IC50 > 18700 nM T20251 CCQ8O9 11567495 IC50 = 4300 nM T20251 CZMB92 11567596 IC50 = 2900 nM T20251 CP7W6H 11567952 IC50 = 4300 nM T20251 CJ3FH6 11568363 IC50 = 80 nM T20251 C52PDV 11568714 IC50 = 3162.28 nM T20251 CMFZ35 11568741 IC50 = 10000 nM T20251 CNV08X 11569158 IC50 = 14000 nM T20251 C0J3VR 11569300 IC50 = 2.5 nM T20251 CU6EY8 11569996 IC50 = 1000 nM T20251 CB59HM 11570626 IC50 > 10000 nM T20251 CZD62R 11572546 Ki = 8000 nM T20251 C18BAJ 11572597 IC50 = 27700 nM T20251 C12VCK 11573765 IC50 = 20000 nM T20251 CMX60P 11573849 IC50 > 6870 nM T20251 C3UQL8 11573971 IC50 = 3500 nM T20251 C86YFM 11575878 IC50 < 25118.86 nM T20251 CFC7D3 11576079 IC50 = 9000 nM T20251 CTVX46 11576269 IC50 > 10000 nM T20251 CASH81 11576387 IC50 = 1258.93 nM T20251 C8JW7U 11577059 IC50 = 11000 nM T20251 C8YLD3 11577158 IC50 = 3162.28 nM T20251 CN87ZF 11577588 IC50 = 1550 nM T20251 CR8E2F 11578028 IC50 = 3162.28 nM T20251 CXP2M0 11580426 Ki > 5000 nM T20251 CW7G3X 11580427 Ki > 5 nM T20251 C7I5KM 11581252 Ki = 5200 nM T20251 CE0U8J 11581337 IC50 = 2900 nM T20251 CN1I8D 11581636 IC50 = 6300 nM T20251 CZ28HJ 11581919 IC50 = 6600 nM T20251 CICM46 11582059 Ki = 1600 nM T20251 CVIP95 11582321 IC50 = 2000 nM T20251 C2DG4A 11582651 IC50 = 930 nM T20251 CM0H2R 11583049 IC50 = 6.2 nM T20251 CZ6C8H 11583193 IC50 = 51100 nM T20251 CP53LK 11583743 IC50 > 10000 nM T20251 CP07QN 11583835 IC50 = 450 nM T20251 C0HFP7 11584185 IC50 = 398.11 nM T20251 C6D1MA 11584660 IC50 = 1995.26 nM T20251 CU4J2W 11584694 IC50 = 31.62 nM T20251 CN5DQ9 11585034 IC50 = 2511.89 nM T20251 C73UHS 11585248 IC50 = 1584.89 nM T20251 CR78YS 11585375 IC50 < 1200 nM T20251 CY3A4K 11587772 IC50 = 2270 nM T20251 C5JBF8 11589054 IC50 < 25118.86 nM T20251 COE14C 11589812 IC50 = 6080 nM T20251 CA2KX0 11590078 IC50 > 10000 nM T20251 C7A3OZ 11590444 IC50 < 31622.78 nM T20251 CC75MD 11590828 IC50 = 3981.07 nM T20251 CK4E6V 11591222 IC50 = 12000 nM T20251 CYX50J 11591601 IC50 = 1000 nM T20251 CIUL60 11591633 IC50 = 251.19 nM T20251 CD6Y3F 11592099 IC50 = 11000 nM T20251 C47TZG 11595633 IC50 = 14000 nM T20251 C1A3PZ 11595635 IC50 = 31600 nM T20251 CMAF85 11596311 IC50 = 9.8 nM T20251 COS24N 11596426 IC50 = 8100 nM T20251 C5NRD9 11596521 Ki = 390 nM T20251 CAU85E 11597758 IC50 = 2400 nM T20251 C3LO6F 11597868 IC50 = 7079.46 nM T20251 CH0OD8 11598084 IC50 < 300 nM T20251 C1TOP5 11598123 IC50 = 2511.89 nM T20251 C6KVY0 11598137 IC50 = 9600 nM T20251 CP56DO 11599295 IC50 > 10000 nM T20251 CKI9D5 11599973 IC50 > 31600 nM T20251 CY72UC 11602409 IC50 > 1500 nM T20251 C1GL6E 11602780 IC50 = 3698.63 nM T20251 C7T3WI 11603194 Ki = 480 nM T20251 CRDU82 11603367 IC50 = 11600 nM T20251 C8GVH9 11603554 IC50 = 22387.21 nM T20251 C04ORX 11603648 Ki = 5000 nM T20251 CPXV24 11603996 IC50 > 100000 nM T20251 CH4AE5 11604196 Ki = 6400 nM T20251 C3V9LT 11604824 IC50 = 70000 nM T20251 COI0G2 11605470 Ki = 89 nM T20251 C9DI6R 11606176 IC50 = 19952.62 nM T20251 CO1A5Z 11606378 IC50 = 2511.89 nM T20251 CL04ZJ 11606435 IC50 = 1000 nM T20251 CJC5N8 11606456 IC50 = 3981.07 nM T20251 C83DCU 11609760 IC50 = 2800 nM T20251 C6HLN8 11610150 IC50 = 2810 nM T20251 CC5R1Q 11610423 Ki = 200 nM T20251 CAU61Q 11610483 IC50 = 3550 nM T20251 CD2PU0 11610816 IC50 > 10000 nM T20251 CTF7J8 11611218 IC50 > 30000 nM T20251 COW93C 11611844 IC50 > 63000 nM T20251 C1WI4H 11611859 IC50 = 6100 nM T20251 CZ4B9T 11612643 IC50 = 7500 nM T20251 C6LUG4 11612700 IC50 > 10000 nM T20251 CT16JP 11613587 IC50 = 199.53 nM T20251 CQL5S8 11613750 IC50 = 16000 nM T20251 CN91SZ 11613873 IC50 = 2511.89 nM T20251 C3FQP1 11614515 IC50 = 2100 nM T20251 C8JAM4 11616357 Ki = 12000 nM T20251 CD28IH 11618024 IC50 = 5600 nM T20251 CA5W9R 11618060 EC50 = 9000 nM T20251 C36OSA 11618702 IC50 = 1100 nM T20251 C1GB6K 11618861 Ki = 1500 nM T20251 CA6X1R 11619076 IC50 < 25118.86 nM T20251 CG1RP5 11619850 IC50 = 1.4 nM T20251 CJ73BI 11619909 IC50 = 10000 nM T20251 CKB59U 11620847 IC50 = 3981.07 nM T20251 CXY07A 11621352 IC50 = 251.19 nM T20251 C79OMR 11623756 Ki > 5 nM T20251 C1KD4Z 11623823 IC50 = 40200 nM T20251 CSB9O5 11623845 Ki > 5000 nM T20251 CD2H3T 11624832 IC50 = 18000 nM T20251 C9WMX4 11624970 IC50 = 500 nM T20251 CX1M6Z 11625277 IC50 = 1800 nM T20251 C34OQC 11626062 IC50 = 1000 nM T20251 C6EGB7 11626833 IC50 = 54000 nM T20251 C7C8FX 11626984 Ki = 42 nM T20251 CIO53A 11627085 IC50 > 31600 nM T20251 C3CP2G 11627368 IC50 > 3200 nM T20251 C9FSA8 11627847 IC50 = 1995.26 nM T20251 C51IBH 11627879 IC50 = 5011.87 nM T20251 CEK0Z8 11628328 IC50 > 31600 nM T20251 CE8W1Z 11628452 IC50 = 501.19 nM T20251 CFJN71 11628631 IC50 = 100 nM T20251 C95RDI 11631662 IC50 > 30000 nM T20251 C0G6PN 11632103 IC50 > 10000 nM T20251 CPV49C 11632254 IC50 = 1000 nM T20251 CNS5P7 11632418 IC50 = 1600 nM T20251 C9HCM6 11632711 Ki = 340 nM T20251 CK34LS 11632737 IC50 = 16600 nM T20251 C7H0AV 11633028 Ki = 1500 nM T20251 C1R2BZ 11633045 IC50 = 12600 nM T20251 CWE63G 11633344 IC50 < 25118.86 nM T20251 CD83GL 11634069 IC50 = 36000 nM T20251 CJBR83 11634073 IC50 = 17000 nM T20251 COB0P4 11634166 Ki = 5100 nM T20251 CO68YB 11634336 IC50 = 31000 nM T20251 CYL45U 11634544 IC50 > 10000 nM T20251 C52ZKM 11634651 IC50 > 10000 nM T20251 C75FNR 11634886 IC50 = 1730 nM T20251 CDE1G8 11635187 IC50 > 31600 nM T20251 C8Y9AL 11635230 IC50 > 31600 nM T20251 CUN3R9 11635332 IC50 > 31600 nM T20251 C23XSL 11638166 Ki = 1800 nM T20251 CCE90V 11638319 IC50 > 60000 nM T20251 CQ1U9W 11638962 IC50 = 7570 nM T20251 COLF16 11639342 IC50 = 213000 nM T20251 CR5QB1 11640354 Ki = 930 nM T20251 CIMW51 11640376 Ki = 3800 nM T20251 CY3IN5 11640515 IC50 = 8300 nM T20251 CMNV51 11640588 Ki = 400 nM T20251 CI2KZ1 11641036 IC50 = 170 nM T20251 CWHK19 11641315 IC50 = 11000 nM T20251 C0XC2N 11641596 IC50 = 3981.07 nM T20251 C25KGE 11641641 IC50 = 251.19 nM T20251 C8DXS0 11642163 IC50 = 794.33 nM T20251 CSE96X 11645396 Ki = 3000 nM T20251 CDP23M 11645473 IC50 = 6400 nM T20251 C0M9NX 11646364 Ki = 2100 nM T20251 CW42YV 11646372 IC50 = 7400 nM T20251 CLR3P8 11646541 IC50 = 10000 nM T20251 C24DVX 11647025 Ki = 2600 nM T20251 C9IOM8 11647276 IC50 = 1300 nM T20251 CJQK24 11647458 IC50 = 34600 nM T20251 C6Y4HR 11647548 IC50 > 30000 nM T20251 CPO25R 11647576 IC50 = 4000 nM T20251 C83VLD 11648483 Ki = 1200 nM T20251 CYQB50 11648990 IC50 = 794.33 nM T20251 C0WAT8 11649549 IC50 = 42000 nM T20251 CXG1B4 11649741 IC50 > 100000 nM T20251 CZPG34 11650178 IC50 > 10000 nM T20251 CM5PG0 11653478 Ki = 10000 nM T20251 CEXK54 11653686 IC50 = 15190 nM T20251 C8I7UT 11654412 IC50 = 9 nM T20251 C2R9QT 11654739 Ki = 300 nM T20251 CGU87J 11654962 IC50 = 6300 nM T20251 C0EF3I 11655513 IC50 = 36900 nM T20251 CPH9X5 11655664 IC50 = 4100 nM T20251 CX7FR8 11655728 IC50 > 10000 nM T20251 C48HCV 11656243 IC50 = 2511.89 nM T20251 CVY3H4 11656753 IC50 = 5610 nM T20251 CPE83G 11656848 IC50 = 1258.93 nM T20251 CT14BC 11657494 IC50 = 251.19 nM T20251 CH3N1I 11659592 IC50 = 490 nM T20251 CF92SM 11659664 IC50 = 24700 nM T20251 CC36GP 11660512 Ki = 10000 nM T20251 CR92TH 11660563 IC50 = 3450 nM T20251 CN6Y7D 11661294 IC50 = 7900 nM T20251 C4G9CM 11661358 IC50 > 10000 nM T20251 CMC02O 11661752 Ki = 8700 nM T20251 CXPC31 11662060 IC50 > 100000 nM T20251 CEL15N 11662194 IC50 > 63095.73 nM T20251 C1F9VA 11662657 IC50 = 15600 nM T20251 CKP76R 11662966 IC50 = 10000 nM T20251 CT2AZ4 11663315 Ki = 380 nM T20251 CBU0L8 11663504 IC50 = 5011.87 nM T20251 C69RQX 11663526 IC50 = 2511.89 nM T20251 C3SJO5 11663578 IC50 = 794.33 nM T20251 C1PB0O 11663999 IC50 = 1258.93 nM T20251 C16UWH 11664328 IC50 = 5011.87 nM T20251 CO15KF 11664409 IC50 > 10000 nM T20251 CG3W2T 11666681 Ki = 31000 nM T20251 CPW3A8 11667985 IC50 = 6600 nM T20251 CJSN27 11668594 IC50 = 3000 nM T20251 C64GUF 11668827 Ki = 7900 nM T20251 CFEQ23 11669001 Ki = 5100 nM T20251 C5SJ9K 11669355 Ki = 700 nM T20251 CNE2K5 11669953 IC50 = 25118.86 nM T20251 CU9P5O 11670029 Ki = 900 nM T20251 CPVR45 11670647 IC50 = 794.33 nM T20251 CE6A2S 11671079 IC50 = 780 nM T20251 CX1GS0 11672017 IC50 = 1220 nM T20251 CON70D 11672049 IC50 = 7900 nM T20251 CT3BP5 11674529 IC50 > 10000 nM T20251 CD9XU6 11675152 IC50 < 25118.86 nM T20251 C7A0WS 11675333 IC50 > 10000 nM T20251 C0V7SU 11675388 IC50 = 5235 nM T20251 C29PWK 11675645 IC50 = 1300 nM T20251 CXB59V 11676220 IC50 = 1.7 nM T20251 CX04MA 11676364 IC50 > 150000 nM T20251 CFQP90 11676381 Ki = 62 nM T20251 C3US8X 11676399 Ki = 720 nM T20251 CY5UB8 11676600 Ki = 260 nM T20251 C6GVU2 11676790 IC50 = 31600 nM T20251 CWQ3M4 11677768 IC50 = 1584.89 nM T20251 C6C4BJ 11678080 IC50 = 1995.26 nM T20251 C34RDZ 11678857 Ki = 364 nM T20251 C7JVX2 11681378 Ki > 5000 nM T20251 C7T9ES 11681588 IC50 = 27000 nM T20251 C8RA5V 11682068 IC50 > 10000 nM T20251 C2JSO8 11683474 IC50 < 31622.78 nM T20251 CEHG64 11683903 IC50 = 15.9 nM T20251 CI6JR2 11684405 IC50 = 6300 nM T20251 C1ZD6V 11685267 IC50 = 1258.93 nM T20251 C9K3EO 11688027 IC50 > 60000 nM T20251 CY36RI 11688223 IC50 = 220 nM T20251 CD1O9I 11688761 IC50 > 1000 nM T20251 C87TCD 11689687 IC50 = 1700 nM T20251 C6S2GN 11689802 IC50 = 400 nM T20251 CR91QA 11690139 IC50 = 5000 nM T20251 CRXO13 11690171 Ki = 1200 nM T20251 CG13YQ 11691697 IC50 = 1258.93 nM T20251 CE1KI3 11692214 IC50 = 501.19 nM T20251 CKX65Z 11692293 IC50 = 66000 nM T20251 CGM36K 11692376 IC50 = 1584.89 nM T20251 C7Z0SX 11695591 IC50 = 2300 nM T20251 CFGR63 11695646 IC50 = 15000 nM T20251 CP3G0Q 11695811 IC50 = 1800 nM T20251 CLT3Z7 11695929 EC50 = 5000 nM T20251 CWX2F0 11696319 IC50 = 940 nM T20251 C8QIH0 11696657 IC50 = 2000 nM T20251 CDV58J 11696813 Ki = 930 nM T20251 CX7MT8 11697412 Ki = 500 nM T20251 C8K3OV 11698389 Ki = 150 nM T20251 CT5J9M 11699340 IC50 = 1584.89 nM T20251 CFCB20 11699532 IC50 = 316.23 nM T20251 C4DJ1V 11699804 IC50 > 10000 nM T20251 CBDC74 11702114 IC50 = 590 nM T20251 CQ5P2F 11702115 IC50 = 890 nM T20251 CXFK83 11702578 Ki > 5000 nM T20251 CZ9SY1 11702625 IC50 = 75000 nM T20251 C5UEI7 11703527 Ki = 320 nM T20251 C9SX7H 11704191 Ki = 13000 nM T20251 C3XDB2 11704592 IC50 = 4100 nM T20251 CTZ61B 11704809 IC50 > 95000 nM T20251 CGD80W 11705119 IC50 = 5011.87 nM T20251 CH5B6O 11705343 IC50 = 32000 nM T20251 C2E8BF 11705395 Ki = 30 nM T20251 CLK68A 11705570 IC50 = 1995.26 nM T20251 CPC67X 11705929 IC50 = 501.19 nM T20251 CG2LE3 11706442 IC50 = 3800 nM T20251 CE1FU8 11706443 IC50 = 2300 nM T20251 C04VLB 11706579 Ki > 10000 nM T20251 CG0B5Q 11706981 IC50 = 3300 nM T20251 C3M8DW 11709098 IC50 = 16200 nM T20251 CXMH25 11710453 Ki = 2000 nM T20251 C4M9AU 11710505 IC50 = 2950 nM T20251 CK1FB9 11710573 IC50 < 25118.86 nM T20251 C12EZH 11710694 Ki = 10000 nM T20251 C5FZ1J 11710873 Ki = 3000 nM T20251 C6CM7S 11711078 IC50 = 7900 nM T20251 CIZQ65 11711452 IC50 = 5280 nM T20251 CIUV17 11711973 IC50 = 800 nM T20251 CN8FE3 11712044 IC50 = 15848.93 nM T20251 C9WI7N 11712071 IC50 = 8317.64 nM T20251 CLY3T0 11712237 IC50 = 8000 nM T20251 C5RZ3S 11712530 Ki = 200 nM T20251 CL3H6E 11712583 IC50 = 1200 nM T20251 CHK5I2 11712756 IC50 = 1584.89 nM T20251 C8V9XO 11712898 IC50 = 560 nM T20251 CWQ67V 11713742 IC50 = 9180 nM T20251 C1XYK2 11717025 IC50 = 17000 nM T20251 CI1C4Z 11718272 Ki = 400 nM T20251 C74DRE 11719291 IC50 = 85500 nM T20251 C9R0FW 11719590 IC50 > 10000 nM T20251 CO29BN 11719912 IC50 = 3080 nM T20251 CD9A0J 11720104 IC50 > 10000 nM T20251 C3FP8J 11720191 IC50 = 5600 nM T20251 CX9VH0 11720815 IC50 = 1000 nM T20251 CXUM63 11720838 IC50 = 794.33 nM T20251 C37DMH 11721190 IC50 = 794.33 nM T20251 CIH38K 11723422 Ki = 10000 nM T20251 CP7EV6 11731453 Ki = 21000 nM T20251 CB8N9K 11732098 IC50 = 11000.01 nM T20251 CA7FS4 11732896 IC50 = 2600 nM T20251 CT23IZ 11742071 IC50 = 6.918 nM T20251 CM95SZ 11744578 Ki = 530 nM T20251 CG0YB2 11751828 IC50 = 390 nM T20251 C4L9EC 11752457 IC50 = 24000 nM T20251 C41OBD 11756414 IC50 = 4000 nM T20251 CKW9D4 11756884 IC50 = 17000 nM T20251 C58DMZ 11757696 IC50 = 3200 nM T20251 CZ8E3X 11771731 IC50 < 1000 nM T20251 C7JD4S 11775505 IC50 = 10.5 nM T20251 C5QGC3 11775544 IC50 = 3162.28 nM T20251 CHS9Q3 11785237 IC50 = 5000 nM T20251 CD13QV 11786769 IC50 = 2800 nM T20251 COB43E 11825520 Ki = 150 nM T20251 CG6Q1B 11842628 IC50 = 19700 nM T20251 CD0F5T 11842667 IC50 = 15135.61 nM T20251 CBC08P 11846124 IC50 > 100000 nM T20251 C5LIW2 11846126 IC50 > 100000 nM T20251 CAD8P9 11848624 IC50 < 100 nM T20251 CCT5G7 11848677 IC50 = 3500 nM T20251 CL6B5X 11848835 IC50 = 430 nM T20251 C3UQT0 11853349 IC50 = 2000 nM T20251 C8VK4D 11853588 IC50 = 13000 nM T20251 CYLO43 11854292 Ki = 1900 nM T20251 C1YD8G 11857777 IC50 = 954992586 nM T20251 CXLW54 11948707 Ki > 10000 nM T20251 CP79ZF 11949710 IC50 = 3900 nM T20251 CQSU51 11950826 IC50 = 14125.38 nM T20251 C85VJZ 11950827 IC50 = 1905.46 nM T20251 CQVX45 11950828 IC50 = 208.93 nM T20251 C0WVX4 11951000 IC50 = 8511.38 nM T20251 C0HT7M 11951722 IC50 = 28000 nM T20251 CTR9Z0 11951723 IC50 = 14200 nM T20251 C4EVI9 11951724 IC50 > 30000 nM T20251 CFYK69 11951728 IC50 = 2700 nM T20251 C5M9VQ 11951901 IC50 > 31600 nM T20251 C0GLF5 11952264 IC50 = 11600 nM T20251 CJLB31 11952265 IC50 = 7700 nM T20251 C4JE5Y 11952437 IC50 = 4100 nM T20251 CS3FO8 11952438 IC50 = 6700 nM T20251 CB0LK9 11952439 IC50 = 2400 nM T20251 CK13QD 11953409 IC50 = 6000 nM T20251 C8SZH2 11965686 IC50 = 1995.26 nM T20251 C38ACD 11973711 Ki = 107 nM T20251 CA54WB 11973799 IC50 = 5.4 nM T20251 C09SBY 11973800 IC50 = 21.2 nM T20251 C4G3JS 11973801 IC50 = 14.7 nM T20251 CJ51DI 11973802 IC50 = 47.7 nM T20251 C68TIS 11974129 IC50 = 63.7 nM T20251 CU3J7M 11974130 IC50 = 7.4 nM T20251 CN38YH 11974131 IC50 = 5 nM T20251 C5W7EA 11974229 IC50 = 5.6 nM T20251 C3C2EN 11974230 IC50 = 12.2 nM T20251 CAN81B 11974231 IC50 = 10.4 nM T20251 CNCP71 11974346 IC50 = 20.3 nM T20251 C7W6UZ 11975326 IC50 = 6.7 nM T20251 C3EU8T 11975438 IC50 = 19.9 nM T20251 CN5W3V 11978858 Ki = 10000 nM T20251 C1O8ZJ 11983278 Ki > 9000 nM T20251 CHC85I 11983362 IC50 = 34000 nM T20251 CZ9FS3 11990142 Ki > 9000 nM T20251 C0KM5I 11992827 IC50 = 4500 nM T20251 C56OSH 11995342 IC50 = 21877.62 nM T20251 C0SMQ3 11995420 IC50 = 135000 nM T20251 C9KSG8 11995421 IC50 = 16000 nM T20251 CEYB03 11995422 IC50 > 30000 nM T20251 C58BPD 11995424 IC50 = 21000 nM T20251 CTYE90 11995521 IC50 = 10000 nM T20251 C0DE5H 11995522 IC50 = 76000 nM T20251 CR4YS2 11996303 IC50 = 794.33 nM T20251 C7D1AY 11996304 IC50 = 1258.93 nM T20251 C1A2IB 12001199 IC50 = 1584.89 nM T20251 CNO57E 12001832 IC50 > 50118.72 nM T20251 C1QBK8 12094039 IC50 = 9800 nM T20251 C4CE8D 12111141 Ki = 4000 nM T20251 C5P6ND 12429371 IC50 = 1608 nM T20251 CZ1V4O 12896968 IC50 = 1120 nM T20251 CCS5B1 12951762 IC50 = 506 nM T20251 C7BE0Q 12991318 IC50 = 31600 nM T20251 CM6IO1 14645090 Ki = 24 nM T20251 CIJA82 14645095 Ki = 1.6 nM T20251 C3S8RY 14793784 IC50 = 163.9 nM T20251 C0TO1Z 14921509 IC50 = 17 nM T20251 C0I8GC 14985965 IC50 = 190 nM T20251 CE78SG 15006442 IC50 = 10 nM T20251 C8BF2P 15254720 IC50 = 199.53 nM T20251 C60TVD 15392306 Ki = 3900 nM T20251 C9ZO7G 15604796 IC50 = 19300 nM T20251 CCDX50 15940498 IC50 > 50000 nM T20251 C8JIP7 15940801 IC50 = 16000 nM T20251 CBE59I 15940927 Ki = 5800 nM T20251 CTH2A9 15941083 IC50 = 8400 nM T20251 CF30UM 15941086 IC50 = 10800 nM T20251 CM10PF 15941255 IC50 = 300 nM T20251 CHFW18 15942650 IC50 = 35000 nM T20251 CB8H6M 15947119 IC50 = 250 nM T20251 CPD3V1 15949508 IC50 = 4800 nM T20251 CLD0M2 15949839 IC50 = 33000 nM T20251 CUS3W4 15950258 IC50 = 25000 nM T20251 CM63YP 15950387 IC50 = 14000 nM T20251 C9KJ6D 15950538 IC50 > 80000 nM T20251 C4S7AB 15950540 IC50 > 80000 nM T20251 C3U1VO 15950542 IC50 > 80000 nM T20251 CKX8M6 15950615 IC50 > 80000 nM T20251 C2ZYA6 15951338 IC50 = 39000 nM T20251 C1Q8IV 15951410 IC50 = 23000 nM T20251 C8IJ0O 15952316 IC50 = 1300 nM T20251 CWZM24 15953526 IC50 = 13400 nM T20251 CSA02I 15979148 IC50 = 2778 nM T20251 CBE54Y 15979149 IC50 = 5312 nM T20251 C9QO8U 15979276 IC50 > 10000 nM T20251 C3W8ZL 15981007 IC50 = 290 nM T20251 C8VYW0 15981180 IC50 = 10100 nM T20251 CE4VG5 15981891 IC50 = 24300 nM T20251 C3L4HO 15981894 IC50 = 14800 nM T20251 CB76UT 15981895 IC50 = 49100 nM T20251 C5UOH2 15982018 IC50 = 20000 nM T20251 CI1SK2 15982019 IC50 > 100000 nM T20251 CXD9I3 15982149 IC50 = 50700 nM T20251 CX3M7T 15982150 IC50 > 100000 nM T20251 CP3N4C 15982151 IC50 = 42000 nM T20251 CS9N5F 15982407 IC50 = 40000 nM T20251 CAB1P3 15982533 IC50 = 19000 nM T20251 CD34SB 15982534 IC50 = 35000 nM T20251 CG50BK 15983304 IC50 = 44000 nM T20251 C5OY3I 15983430 IC50 = 29000 nM T20251 CBE59Y 15983549 IC50 = 13000 nM T20251 C6YAJ0 15983550 IC50 = 12900 nM T20251 CUX86I 15983552 IC50 = 6000 nM T20251 CO02BA 15983553 IC50 = 9000 nM T20251 C9TO6J 15983677 IC50 = 3000 nM T20251 CIV82J 15983679 IC50 = 41000 nM T20251 C30OTX 15983680 IC50 = 1400 nM T20251 CT2G7E 15983809 IC50 = 2800 nM T20251 C0GMT8 15983810 IC50 > 100000 nM T20251 CPR25X 15986917 IC50 < 31622.78 nM T20251 CRBP36 15987008 IC50 = 6309.57 nM T20251 C5KW3L 15987108 IC50 = 9332.54 nM T20251 CF6S2D 15987282 IC50 < 63095.73 nM T20251 CXU15Z 15987451 IC50 = 7943.28 nM T20251 C6V3WY 15987452 IC50 < 15848.93 nM T20251 C0HKS9 16004748 IC50 > 10000 nM T20251 CV0YA4 16005493 IC50 = 8410 nM T20251 CG8KR9 16005860 IC50 = 4114 nM T20251 C70KBE 16006079 IC50 = 2220 nM T20251 CCL59Z 16007088 IC50 = 1900 nM T20251 CG5A7W 16013152 IC50 > 30000 nM T20251 CBMF65 16013184 IC50 > 30000 nM T20251 C6V4TG 16013186 IC50 > 30000 nM T20251 CUB5X2 16038385 IC50 > 63095.73 nM T20251 C8AB4L 16039796 IC50 = 18000 nM T20251 CA7QW1 16039834 IC50 = 40000 nM T20251 CPCZ62 16040329 IC50 = 19000 nM T20251 C20CRP 16040587 IC50 > 31622.78 nM T20251 CH8K6G 16040671 IC50 = 31622.78 nM T20251 C8ZP3G 16041292 IC50 > 25118.86 nM T20251 CDU1L0 16041411 IC50 > 30000 nM T20251 CGM4N8 16041594 IC50 > 40000 nM T20251 C1V9EY 16041612 IC50 > 10000 nM T20251 CX9W7Q 16043220 IC50 = 690 nM T20251 CJ78MO 16045297 Ki = 31622.78 nM T20251 CB64EN 16049818 IC50 > 30000 nM T20251 CU27FI 16049886 IC50 = 156666.67 nM T20251 CZC7L2 16049887 IC50 = 115000 nM T20251 CQ9U1Y 16051921 IC50 = 2400 nM T20251 CS8NZ0 16059780 Ki = 6200 nM T20251 C6V4HS 16059786 IC50 = 440 nM T20251 CC2YJ8 16062553 IC50 > 10000 nM T20251 C1LH5T 16062816 IC50 > 10000 nM T20251 C7UCS5 16064456 Ki > 20000 nM T20251 CEZI54 16064872 IC50 = 37153.52 nM T20251 C0V9RI 16064896 Ki > 20000 nM T20251 CM1V6L 16064897 Ki > 20000 nM T20251 C96FEP 16065425 IC50 = 20892.96 nM T20251 CVCJ16 16065428 IC50 = 7762.47 nM T20251 C6MC0Z 16065567 IC50 = 30199.52 nM T20251 CPN9H5 16065569 IC50 = 16595.87 nM T20251 CL1M3W 16065704 IC50 = 16595.87 nM T20251 CF3UG1 16066664 IC50 = 1100 nM T20251 C30UFT 16066811 Ki > 30000 nM T20251 CI1EC9 16068009 Ki = 17000 nM T20251 C3ZKJ5 16068120 Ki = 4400 nM T20251 CPLU48 16068121 Ki = 3800 nM T20251 C9S6QP 16068233 Ki = 13000 nM T20251 CB9Z0L 16068234 Ki = 2600 nM T20251 CW4U7H 16068235 Ki > 20000 nM T20251 CT4JA5 16068236 Ki > 20000 nM T20251 C8SQ5I 16068237 Ki = 6300 nM T20251 CVT0E7 16070046 Ki = 30000 nM T20251 CZ47FJ 16071018 IC50 = 12589.25 nM T20251 CQ06FD 16071731 IC50 = 28000 nM T20251 C3LK2C 16072132 IC50 = 8100 nM T20251 CBM80K 16091080 IC50 = 5319 nM T20251 CX5KI3 16105788 Ki > 10000 nM T20251 CKPQ93 16112836 IC50 = 1584.89 nM T20251 CZC0H1 16116961 IC50 = 25000 nM T20251 CYV05C 16123136 IC50 = 1000 nM T20251 C8C2IW 16123138 IC50 = 100 nM T20251 C7YF8I 16123140 IC50 = 1258.93 nM T20251 C91DQN 16123241 IC50 = 1584.89 nM T20251 CQG7P8 16123247 IC50 = 1258.93 nM T20251 CA6D4S 16123347 IC50 = 1258.93 nM T20251 CBH5P4 16123349 IC50 = 794.33 nM T20251 CPN48R 16123353 IC50 = 1995.26 nM T20251 CK7H2W 16123462 IC50 = 1258.93 nM T20251 C5MY2Q 16123464 IC50 = 10000 nM T20251 CNQ6J2 16123467 IC50 = 3162.28 nM T20251 CWU6P3 16123945 IC50 = 25118.86 nM T20251 CZF23I 16124479 Ki > 100000 nM T20251 C9G8TZ 16124598 IC50 > 31622.78 nM T20251 CYI7J5 16126731 Ki = 16 nM T20251 CTRP20 16190907 IC50 = 15500 nM T20251 CK8Z9L 16220221 IC50 = 2750 nM T20251 CFI8G2 16220223 IC50 = 5300 nM T20251 CTU7J0 16220225 IC50 > 10000 nM T20251 C0ZUH7 16220280 IC50 = 1800 nM T20251 C39SIQ 16220281 IC50 > 10000 nM T20251 C0JA4Q 16220791 IC50 = 5190 nM T20251 CWIT69 16220793 IC50 = 450 nM T20251 CI84RL 16220795 IC50 = 790 nM T20251 C3W1LK 16220874 IC50 = 2590 nM T20251 CUNW89 16220876 IC50 = 3590 nM T20251 C1VUC5 16220877 IC50 = 2500 nM T20251 CN91VO 16220879 IC50 = 3390 nM T20251 CVQ9T5 16220880 IC50 = 4800 nM T20251 C1U9XM 16220882 IC50 = 1750 nM T20251 CZUQ73 16220957 IC50 = 7460 nM T20251 CA5NX6 16220959 IC50 = 1740 nM T20251 C8J3YN 16220960 IC50 = 5870 nM T20251 CPV4G2 16220962 IC50 = 80 nM T20251 C4L7QD 16221024 IC50 = 2100 nM T20251 CAU7E0 16221025 IC50 > 10000 nM T20251 C4GPA2 16221027 IC50 = 1720 nM T20251 C3SH0K 16221088 IC50 > 10000 nM T20251 CM8N1R 16221090 IC50 > 10000 nM T20251 C5E6AC 16221091 IC50 = 1430 nM T20251 CXL6V8 16221092 IC50 > 10000 nM T20251 CW35VX 16221140 IC50 = 1700 nM T20251 C78VJQ 16221258 IC50 = 4870 nM T20251 C9X2GY 16221259 IC50 = 7910 nM T20251 CIA5Y4 16221343 IC50 > 30000 nM T20251 C3P7XC 16221373 IC50 > 10000 nM T20251 CJ8RC1 16221375 IC50 = 53000 nM T20251 C5TV3A 16221425 IC50 > 10000 nM T20251 C8CKV2 16221426 IC50 > 10000 nM T20251 CQE9N1 16221427 IC50 = 2560 nM T20251 CS8W9L 16222361 Ki = 794.33 nM T20251 C2UV9Y 16222392 IC50 > 30000 nM T20251 CA20NM 16222570 Ki = 19952.62 nM T20251 CTH6W4 16292141 IC50 > 25000 nM T20251 CHAY38 16352480 IC50 = 25118.86 nM T20251 CP71ZQ 16389349 IC50 > 50118.72 nM T20251 CX57MU 16648749 IC50 = 6770 nM T20251 C4QU0M 16654984 IC50 = 1200 nM T20251 C6P4BX 16656803 IC50 = 1510 nM T20251 C23NUI 16659197 IC50 = 30000 nM T20251 COC0B8 16659239 IC50 = 25000 nM T20251 CIBY49 16661548 IC50 = 2800 nM T20251 CU9LS2 16661702 IC50 = 780 nM T20251 CYF7U1 16662313 IC50 > 30000 nM T20251 CS90PN 16718565 IC50 = 12600 nM T20251 C7K5AW 16721015 IC50 = 7870 nM T20251 CS14WU 16722242 IC50 > 30000 nM T20251 C8T4JF 16722295 IC50 = 128000 nM T20251 CW62MC 16725327 IC50 = 23000 nM T20251 C4YMP1 16725956 Ki = 206 nM T20251 C92NRU 16727109 IC50 > 80000 nM T20251 COJU37 16727124 IC50 = 200 nM T20251 C4U5XO 16730656 Ki = 18 nM T20251 C8KRM1 16730814 Ki = 4710 nM T20251 C2CRF5 16730815 Ki > 10000 nM T20251 C1D5EW 16733141 Ki = 0.39 nM T20251 CR3W5J 16733265 Ki = 980 nM T20251 C5YWS6 16733266 Ki > 1000 nM T20251 CQO3M8 16733807 Ki = 282 nM T20251 CVI8T4 16735967 IC50 = 27500 nM T20251 CV9US5 16736978 IC50 = 8300 nM T20251 CDG57C 16737679 IC50 = 17000 nM T20251 CHU72I 16738321 IC50 = 11000 nM T20251 CV5F3P 16739263 IC50 > 100000 nM T20251 C6DS7K 16739334 Ki = 4342 nM T20251 CI7Z6F 16741239 Ki = 84 nM T20251 CW2SY5 16750291 IC50 = 7200 nM T20251 CGP40H 16784276 IC50 > 10000 nM T20251 CP69WV 16955923 IC50 = 3000 nM T20251 C5DKZ8 16956771 IC50 = 8000 nM T20251 CU42ZC 17244953 IC50 < 10000 nM T20251 CU05RG 17748274 IC50 > 90000 nM T20251 CAJ0S2 17754557 EC50 > 30000 nM T20251 CN6IP3 17915602 IC50 = 20300 nM T20251 CBNK23 17963226 IC50 > 10000 nM T20251 C5ZT8C 17963227 IC50 = 316.23 nM T20251 CQ7WR1 17963315 IC50 = 10000 nM T20251 C2V6WP 17963332 IC50 > 10000 nM T20251 COCE85 17963334 IC50 > 10000 nM T20251 C2PWS7 17963363 IC50 = 12589.25 nM T20251 C1DVQ9 18004024 IC50 = 562.34 nM T20251 CV5EG7 18727564 Ki > 10000 nM T20251 C1OE8D 18971393 IC50 > 100000 nM T20251 C9JD5Y 19360456 IC50 = 3500 nM T20251 CCA0T1 19958773 IC50 = 2600 nM T20251 C8ICF9 20111627 IC50 = 4300 nM T20251 CES62Q 20299676 IC50 = 300 nM T20251 CSO6R2 20579370 IC50 = 6680 nM T20251 C5S7YM 20579374 IC50 = 1540 nM T20251 C09RQX 20579375 IC50 = 480 nM T20251 CXM1R3 20579392 IC50 = 1480 nM T20251 CWFZ97 20579393 IC50 = 7450 nM T20251 CQAX57 20579471 IC50 = 5920 nM T20251 CFQM24 20664161 IC50 = 2700 nM T20251 C8WSD5 20747478 Ki = 970 nM T20251 CSV2M0 20817761 Ki = 112 nM T20251 C85YPN 20817762 Ki > 2000 nM T20251 CO29QJ 20817763 Ki > 2000 nM T20251 CS4AU1 20817821 Ki = 215 nM T20251 CZC89U 20817846 Ki = 30 nM T20251 CHB01Q 20817864 Ki = 1440 nM T20251 COR4F2 21031286 IC50 > 10000 nM T20251 CMA0D8 21050485 Ki = 4000 nM T20251 C1CA6D 21070989 IC50 = 16000 nM T20251 CAO91K 21099378 Ki = 4000 nM T20251 C9MDU4 21099413 Ki = 8200 nM T20251 C2LMD4 21099424 Ki > 9000 nM T20251 CJB73F 21099433 Ki > 9000 nM T20251 CQU60A 21099448 Ki = 3300 nM T20251 CBCL34 21099463 Ki > 9000 nM T20251 C36INC 21099465 Ki > 9000 nM T20251 C6GRC9 21099470 Ki = 2800 nM T20251 CY75XP 21099472 Ki = 9000 nM T20251 CCO7D2 21099473 Ki > 9000 nM T20251 CP94VE 21099486 Ki > 9000 nM T20251 CF90PJ 21099505 Ki = 7919 nM T20251 CDBY94 21099514 Ki = 6900 nM T20251 CB12UT 21099515 Ki = 9500 nM T20251 C5JCZ6 21193534 Ki = 500 nM T20251 CN85CQ 21252889 IC50 = 2630 nM T20251 CN1XA4 21252891 IC50 = 32500 nM T20251 C18TEI 21303363 IC50 = 8600 nM T20251 COR3F0 21315851 IC50 = 2790 nM T20251 CJV03C 21347732 IC50 < 30000 nM T20251 C6F8SM 21445141 IC50 = 30 nM T20251 CO17PU 21635104 IC50 = 25118.86 nM T20251 C0R5XN 21949788 IC50 = 39000 nM T20251 CCT37S 21949819 IC50 = 9800 nM T20251 C80SEF 21949901 IC50 = 100000 nM T20251 CU0O4K 21955317 Ki = 260 nM T20251 CSZ30L 21998522 Ki = 36870 nM T20251 CSQ2Y0 22017550 Ki = 1268 nM T20251 CJ76FL 22037373 IC50 > 100000 nM T20251 CE65DB 22115679 Ki = 1280 nM T20251 CO32YX 22254068 IC50 > 10000 nM T20251 C0UMW7 22262550 IC50 = 790 nM T20251 C4NO6Y 22315157 IC50 = 23000 nM T20251 C16HAP 22348022 Ki = 355 nM T20251 CCU37W 22348066 Ki = 420 nM T20251 C82XIL 22348140 Ki = 280 nM T20251 CY0WA7 22348155 Ki = 550 nM T20251 C5PS4N 22348219 Ki > 2000 nM T20251 C6KJ0C 22348261 Ki = 778 nM T20251 CMZH62 22391985 IC50 > 94500 nM T20251 CMV28G 22458335 Ki > 10000 nM T20251 CEB1M3 22724580 Ki = 300 nM T20251 CD14YL 23102733 IC50 = 6309.57 nM T20251 CU1T8V 23102749 IC50 = 3981.07 nM T20251 CYW7Q6 23150305 Ki = 8 nM T20251 C5MXI2 23151144 IC50 = 6800 nM T20251 CCES43 23151160 IC50 > 10000 nM T20251 CX6DW5 23151169 IC50 > 10000 nM T20251 C6QC2D 23151199 IC50 = 7900 nM T20251 CGB8I7 23151202 IC50 = 6400 nM T20251 CY8U0D 23151208 IC50 > 10000 nM T20251 C3BP7D 23151209 IC50 > 10000 nM T20251 CT78IA 23151210 IC50 > 10000 nM T20251 C31KDO 23151223 IC50 = 10000 nM T20251 CQ1K7H 23151224 IC50 = 10000 nM T20251 CU24MC 23151229 IC50 > 10000 nM T20251 CM63GT 23151246 IC50 > 10000 nM T20251 C47RDY 23151248 IC50 > 10000 nM T20251 CU4DK0 23151250 IC50 > 10000 nM T20251 C1D0AE 23151312 IC50 > 10000 nM T20251 CE50PJ 23151323 IC50 > 10000 nM T20251 C2KQ6N 23151327 IC50 > 10000 nM T20251 CGJ78I 23151329 IC50 = 8000 nM T20251 COPR89 23151331 IC50 > 10000 nM T20251 C2NYB8 23151337 IC50 > 10000 nM T20251 C12SUL 23151367 IC50 > 10000 nM T20251 C3TVL7 23501721 IC50 > 3000 nM T20251 C7YFT3 23582127 IC50 = 10300 nM T20251 C5E8TY 23582189 Ki = 18540 nM T20251 CL1YH7 23582308 IC50 = 6309.57 nM T20251 C0EJK3 23585071 IC50 > 32000 nM T20251 CW2R4M 23624283 IC50 = 16982.44 nM T20251 C8VD3S 23624312 IC50 = 5400 nM T20251 CMV89L 23625920 IC50 = 2228.44 nM T20251 CW6OB1 23627212 IC50 > 10000 nM T20251 C0R8OI 23628252 IC50 > 10000 nM T20251 CUI9H4 23630215 IC50 = 1200 nM T20251 CK6B7G 23630497 IC50 = 125.89 nM T20251 CH95VG 23630499 IC50 = 63.1 nM T20251 C2XLN1 23630501 IC50 = 10 nM T20251 C1N5TV 23630503 IC50 = 794.33 nM T20251 C7WZJ0 23630505 IC50 = 1258.93 nM T20251 C4MI9Y 23630602 IC50 = 125.89 nM T20251 C24TDZ 23630604 IC50 = 39.81 nM T20251 CU8D0O 23630606 IC50 = 39.81 nM T20251 CKB1E5 23630796 IC50 = 794.33 nM T20251 CJ81PU 23630797 IC50 = 316.23 nM T20251 CV68XN 23630900 IC50 = 39.81 nM T20251 CD61SO 23630901 IC50 = 501.19 nM T20251 CY2RG1 23630902 EC50 = 120 nM T20251 CTJS17 23630998 IC50 = 316.23 nM T20251 CXVR30 23630999 IC50 = 1995.26 nM T20251 CSAT45 23631000 IC50 = 63.1 nM T20251 C6EO1W 23631001 IC50 = 251.19 nM T20251 CE3AM4 23631091 IC50 = 251.19 nM T20251 C9BMW2 23631092 IC50 = 79.43 nM T20251 CKT7B3 23631093 IC50 = 398.11 nM T20251 CM8U1D 23631172 IC50 = 3981.07 nM T20251 CH2I1P 23631366 IC50 = 25.12 nM T20251 C6YS4P 23631368 IC50 = 794.33 nM T20251 C4TV8X 23631454 IC50 = 25.12 nM T20251 CE40PT 23631458 IC50 = 316.23 nM T20251 C09NTA 23631540 IC50 = 794.33 nM T20251 C83QKW 23631544 IC50 = 158.49 nM T20251 C0RPW8 23631636 IC50 = 19.95 nM T20251 CQIG80 23633343 IC50 > 300000 nM T20251 CU1LK3 23633350 IC50 = 100 nM T20251 CC8JL7 23634277 IC50 = 289000 nM T20251 CVF78O 23634281 IC50 = 4200 nM T20251 CEB67J 23644676 IC50 = 4600 nM T20251 C2Q5IK 23645581 Ki = 49000 nM T20251 C07DVE 23646575 IC50 = 2900 nM T20251 CKSD05 23646576 IC50 = 2600 nM T20251 CUJ0D3 23646577 IC50 = 8300 nM T20251 CZ0QF1 23648867 IC50 > 30000 nM T20251 C7MZX9 23649185 IC50 = 3382.98 nM T20251 CE29IW 23650547 IC50 = 9800 nM T20251 CGI6M2 23658492 IC50 = 6200 nM T20251 CM7C4W 23661708 IC50 = 100000 nM T20251 CO6L9F 23661716 IC50 = 100000 nM T20251 CHR14F 23661718 IC50 = 20300 nM T20251 C9H4WT 23686961 IC50 > 31622.78 nM T20251 CASU54 23696973 IC50 > 31622.78 nM T20251 C9PY4A 23725172 IC50 = 13000 nM T20251 CO01RG 24178536 IC50 = 700 nM T20251 CL4WV2 24180125 IC50 > 10000 nM T20251 CBXC05 24424330 IC50 = 80 nM T20251 CQ0KU9 24738459 Ki = 2060 nM T20251 CC52AB 24743739 IC50 = 4500 nM T20251 CN0A5T 24744322 Ki = 6330 nM T20251 CCPE43 24744323 Ki = 2790 nM T20251 C8RC9P 24744325 Ki > 30000 nM T20251 CC5T6J 24744326 Ki > 30000 nM T20251 CP98HS 24744473 Ki = 3400 nM T20251 CCG05Q 24744793 Ki = 9790 nM T20251 CGS47I 24744797 Ki = 460 nM T20251 C1SDO5 24744977 IC50 > 10000 nM T20251 C0CHJ8 24745269 Ki = 16740 nM T20251 CT2DX6 24745764 Ki = 28500 nM T20251 CVB7J3 24746434 Ki = 790 nM T20251 C8EYH1 24746435 Ki = 21450 nM T20251 C28AWJ 24746436 Ki = 1210 nM T20251 CSA6C8 24746437 Ki = 3810 nM T20251 CRN13C 24748804 IC50 = 31622.78 nM T20251 CTIF10 24748806 IC50 < 63095.73 nM T20251 CMJU59 24748889 IC50 = 39810.72 nM T20251 CB6R3K 24748890 IC50 < 63095.73 nM T20251 C5EQ8T 24748892 IC50 < 63095.73 nM T20251 C1XN4V 24748896 IC50 < 15848.93 nM T20251 CFR1S3 24748988 IC50 = 12589.25 nM T20251 CG43ZS 24748989 IC50 = 12589.25 nM T20251 C96KDH 24748992 IC50 = 19952.62 nM T20251 CH8N1W 24748993 IC50 < 63095.73 nM T20251 CQF29T 24749076 IC50 = 25118.86 nM T20251 CU0GX7 24749078 IC50 = 12589.25 nM T20251 CGD2I7 24749080 IC50 = 31622.78 nM T20251 CKVA89 24749182 IC50 < 63095.73 nM T20251 CRGJ52 24749183 IC50 < 63095.73 nM T20251 C13GRZ 24749184 IC50 < 63095.73 nM T20251 C8ZE6H 24749185 IC50 < 31622.78 nM T20251 CG9I8K 24749186 IC50 < 63095.73 nM T20251 CF8W2P 24749291 IC50 < 63095.73 nM T20251 CTB38H 24749292 IC50 < 63095.73 nM T20251 CET71X 24749293 IC50 = 19952.62 nM T20251 CAE9S7 24749294 IC50 < 63095.73 nM T20251 CKV83Y 24749295 IC50 = 7943.28 nM T20251 C6S0OJ 24749401 IC50 = 25118.86 nM T20251 CWTB59 24749606 IC50 = 63095.73 nM T20251 CHYC87 24749609 IC50 < 63095.73 nM T20251 CY53AF 24749610 IC50 < 63095.73 nM T20251 CT93NP 24749721 IC50 < 63095.73 nM T20251 C7EGL2 24749724 IC50 = 12589.25 nM T20251 CW19JN 24749726 IC50 = 50118.72 nM T20251 CI6W7D 24749841 IC50 = 501.19 nM T20251 CV20EP 24749844 IC50 < 63095.73 nM T20251 CYI79E 24749958 IC50 < 63095.73 nM T20251 CGT53R 24749959 IC50 < 63095.73 nM T20251 C20QND 24749960 IC50 = 31622.78 nM T20251 CSXA65 24749962 IC50 < 63095.73 nM T20251 CNOX23 24750086 IC50 = 3981.07 nM T20251 C1XRY9 24750087 IC50 < 63095.73 nM T20251 C89WKU 24750088 IC50 < 63095.73 nM T20251 C7I4LK 24750278 IC50 = 200 nM T20251 CI0W8A 24755210 IC50 = 19600 nM T20251 CUGR26 24757965 IC50 = 15000 nM T20251 CX79CS 24757966 IC50 > 30000 nM T20251 C25HKJ 24758044 IC50 = 7000 nM T20251 CJ1QB7 24758481 IC50 = 2511.89 nM T20251 C8CWX4 24758715 IC50 = 794.33 nM T20251 CU06GI 24758717 IC50 = 630.96 nM T20251 CPL05Y 24758828 IC50 = 630.96 nM T20251 C7RZ9I 24758830 IC50 = 1258.93 nM T20251 C6JQC4 24758832 IC50 = 6309.57 nM T20251 CBNF87 24758834 IC50 = 1995.26 nM T20251 CGQL10 24758836 IC50 = 1995.26 nM T20251 CGE32Q 24758838 IC50 = 6309.57 nM T20251 CL80CU 24758945 IC50 = 6309.57 nM T20251 C8JQW6 24758947 IC50 = 2511.89 nM T20251 CJL67N 24759089 IC50 > 100000 nM T20251 CDF15M 24759558 IC50 = 8000 nM T20251 C1KQY0 24759785 IC50 = 1500 nM T20251 C6GBU8 24762221 Ki = 3981.07 nM T20251 CJ0C1I 24765309 IC50 > 10000 nM T20251 CBJ9T3 24765959 IC50 > 10000 nM T20251 C7RGV4 24768404 IC50 = 950 nM T20251 CZ4J5K 24768415 IC50 = 285 nM T20251 C4ZRC9 24768418 IC50 = 1670 nM T20251 CI6B4H 24768423 IC50 = 4170 nM T20251 CS0C6Q 24768425 IC50 = 600 nM T20251 CBMC42 24768429 IC50 = 420 nM T20251 CA3UK5 24768431 IC50 = 1860 nM T20251 CG8QK3 24768432 IC50 = 1010 nM T20251 CMT5N1 24768433 IC50 = 650 nM T20251 C6HW8J 24768434 IC50 = 2280 nM T20251 CU7W4F 24768547 IC50 = 7100 nM T20251 CHI83W 24769038 IC50 = 32.7 nM T20251 C0I2HU 24769156 IC50 = 10000 nM T20251 CX8DH1 24769723 IC50 > 30000 nM T20251 CVR27S 24769783 IC50 = 6400 nM T20251 C56EJY 24771419 IC50 = 1600 nM T20251 C6H9WM 24771420 IC50 = 1400 nM T20251 COGS63 24771524 IC50 = 3500 nM T20251 CJ9W6U 24771741 IC50 = 900 nM T20251 CBA2P0 24776663 IC50 = 5300 nM T20251 C4ZP5A 24776667 IC50 > 30000 nM T20251 CTG41H 24778289 IC50 = 5800 nM T20251 C30AKB 24778290 IC50 > 30000 nM T20251 CTDU84 24778294 IC50 = 20200 nM T20251 CHZ16E 24778412 IC50 = 2100 nM T20251 CU9Z8O 24778415 IC50 > 30000 nM T20251 C4C3HR 24780883 IC50 = 5.8 nM T20251 C8ELU9 24782303 IC50 = 7943.28 nM T20251 CJ6SF5 24782306 IC50 = 31622.78 nM T20251 C01UNQ 24782307 IC50 = 3981.07 nM T20251 C7KB8R 24782550 IC50 = 15848.93 nM T20251 C3VF5D 24782552 IC50 = 19952.62 nM T20251 C1BQK0 24782553 IC50 = 3981.07 nM T20251 CSPX91 24782554 IC50 = 15848.93 nM T20251 C7A8DI 24782800 IC50 = 25118.86 nM T20251 C5TOI2 24782801 IC50 = 6309.57 nM T20251 C7FZ2J 24782802 IC50 = 10000 nM T20251 C8S4LC 24782803 IC50 = 3981.07 nM T20251 C4KT6W 24782804 IC50 = 5011.87 nM T20251 C2IXL5 24782805 IC50 = 12589.25 nM T20251 CDEB17 24783056 IC50 = 12589.25 nM T20251 C3J4RX 24785333 IC50 = 15848.93 nM T20251 CMPH82 24785597 IC50 = 7943.28 nM T20251 C7HI4R 24785600 IC50 = 10000 nM T20251 CV7WH3 24785604 IC50 = 12589.25 nM T20251 CTF93A 24785864 IC50 = 7943.28 nM T20251 C1JX7P 24785870 IC50 = 25118.86 nM T20251 CRD90F 24786134 IC50 = 7943.28 nM T20251 C7K1EU 24786138 IC50 = 6309.57 nM T20251 CM2DL3 24795066 IC50 = 11000 nM T20251 CP1WR0 24795070 IC50 < 1000 nM T20251 CUM03S 24798754 IC50 = 23000 nM T20251 CDQ58K 24799187 IC50 = 8700 nM T20251 CTQ59S 24799364 IC50 = 7100 nM T20251 C8LJY2 24799365 IC50 = 80000 nM T20251 CO32ND 24799366 IC50 = 14000 nM T20251 C6X0JS 24799545 IC50 = 6100 nM T20251 CG24KB 24799546 IC50 = 9500 nM T20251 C1QL3V 24799711 IC50 = 9900 nM T20251 CH0Y9J 24800231 IC50 = 13000 nM T20251 C10YFG 24800398 IC50 = 12000 nM T20251 C3FYB5 24800577 IC50 = 16000 nM T20251 C17RDK 24800578 IC50 = 2300 nM T20251 C30UAB 24800743 IC50 = 8400 nM T20251 C6SHG9 24800925 IC50 = 15000 nM T20251 C0L6CF 24800927 IC50 = 28000 nM T20251 CM2K4N 24801101 IC50 = 20000 nM T20251 CP8T1L 24801102 IC50 = 33000 nM T20251 CA8GT1 24801457 IC50 = 6000 nM T20251 CW8GD6 24801458 IC50 = 7400 nM T20251 CE25UP 24801459 IC50 = 33000 nM T20251 CSK49W 24801626 IC50 = 25000 nM T20251 C1NK4A 24801627 IC50 = 12000 nM T20251 C9GK5S 24801792 IC50 = 43000 nM T20251 CWH29M 24801795 IC50 = 7700 nM T20251 C84TEM 24801797 IC50 = 8300 nM T20251 C2AKX9 24804150 IC50 = 158.49 nM T20251 CJ4RO1 24804774 Ki = 794.33 nM T20251 CK84BF 24804775 Ki = 10000 nM T20251 C1Z3OQ 24804941 Ki = 2511.89 nM T20251 C6AE2U 24804942 Ki = 1584.89 nM T20251 C1ZYM4 24804943 Ki = 1258.93 nM T20251 CBS5J4 24804985 IC50 > 100000 nM T20251 CH15KN 24808474 IC50 = 60 nM T20251 C73QEI 24808475 IC50 > 10000 nM T20251 CWE46Z 24810003 IC50 = 3960 nM T20251 C14FOH 24810867 IC50 = 30000 nM T20251 CT53OY 24810870 IC50 = 19000 nM T20251 CL5YW9 24825703 IC50 > 30000 nM T20251 CJSO87 24849206 IC50 > 10000 nM T20251 CEA01P 24852079 IC50 > 30000 nM T20251 CR7X1M 24856034 EC50 = 900 nM T20251 CEW31B 24856362 IC50 > 100000 nM T20251 CB4LY1 24857598 IC50 = 2500 nM T20251 CSR8J4 24857759 IC50 = 13100 nM T20251 C9O5NZ 24857819 IC50 = 1600 nM T20251 CY9W8O 24860300 EC50 = 408000 nM T20251 CIR64L 24860582 IC50 = 24200 nM T20251 CKZ25G 24862861 IC50 = 19000 nM T20251 CRUQ41 24863611 IC50 = 17000 nM T20251 C3UNC4 24864147 IC50 = 20000 nM T20251 CCV9N3 24866867 IC50 = 31000 nM T20251 C4UEM5 24871537 IC50 = 1230 nM T20251 CP2L5B 24871655 IC50 = 4650 nM T20251 C7RE9Q 24872164 IC50 = 122000 nM T20251 C06DKB 24875236 IC50 = 16000 nM T20251 CA18VT 24875749 IC50 = 1400 nM T20251 CGI85O 24875752 IC50 = 3640 nM T20251 CT4EZ5 24875845 IC50 = 1710 nM T20251 CLHP80 24875846 IC50 = 17800 nM T20251 CS0K2J 24875942 IC50 = 1070 nM T20251 CU34QD 24884554 IC50 = 12789.47 nM T20251 CNF2E4 24885663 IC50 = 1411.76 nM T20251 CJO97K 24885890 IC50 = 7344.83 nM T20251 C0FUC5 24886365 IC50 = 3666.67 nM T20251 C5KA0N 24893979 IC50 = 3790 nM T20251 CRAK17 24893993 IC50 = 8200 nM T20251 CNQ6I4 24894028 IC50 = 3100 nM T20251 C5WS6R 24894100 IC50 > 10000 nM T20251 C3C0KP 24894134 IC50 = 500 nM T20251 C2EQR6 24894426 IC50 = 940 nM T20251 CT9EZ4 24894428 IC50 = 1500 nM T20251 CN1E8M 24894430 IC50 = 11000 nM T20251 C9USO6 24894431 IC50 = 11000 nM T20251 C4IDR3 24894531 IC50 > 50000 nM T20251 C2AU5Y 24894647 IC50 = 2300 nM T20251 CC6F9D 24894783 IC50 > 50000 nM T20251 C8ERZ5 24895094 IC50 = 5010 nM T20251 C1N0CZ 24895351 IC50 > 10000 nM T20251 CI2S7Y 24895452 IC50 = 1000 nM T20251 CU31LR 24895550 IC50 > 10000 nM T20251 C2IQ9J 24896791 IC50 > 30000 nM T20251 CJ3W0E 24897476 IC50 = 3100 nM T20251 CI4UX5 24900018 IC50 = 7400 nM T20251 C7J4ZQ 24900259 IC50 = 11000 nM T20251 C2TWC8 24900261 IC50 = 7700 nM T20251 CT8GA0 24901491 IC50 > 10000 nM T20251 CY3C1U 24901492 IC50 = 1300 nM T20251 CC2GE7 24901493 IC50 = 2200 nM T20251 CFM1P2 24901494 IC50 = 2400 nM T20251 CF24OR 24901496 IC50 = 1500 nM T20251 CAUZ61 24901497 IC50 = 11000 nM T20251 C7IQO2 24901498 IC50 = 26400 nM T20251 C7TC3P 24901586 IC50 = 2700 nM T20251 C4YDO0 24901587 IC50 = 500 nM T20251 CENZ09 24901588 IC50 = 9000 nM T20251 C8IP6E 24901589 IC50 = 5000 nM T20251 CSD0O9 24901590 IC50 = 1500 nM T20251 CZEF59 24901591 IC50 = 20000 nM T20251 CRNK57 24901592 IC50 = 30000 nM T20251 C4DN3Q 24905400 IC50 > 100000 nM T20251 CD50AV 24905911 IC50 = 14600 nM T20251 CIXU54 24905912 IC50 = 19200 nM T20251 CTU12K 24905913 IC50 = 13800 nM T20251 CGN65K 24905914 IC50 = 15200 nM T20251 C9OAG1 24906198 IC50 = 16900 nM T20251 C0BP8C 24939244 IC50 = 0.41 nM T20251 CYL4U5 24948945 IC50 = 3900 nM T20251 CQU27P 24948946 IC50 = 1100 nM T20251 CRJ08Z 24948948 IC50 = 6000 nM T20251 CC17EO 24950873 IC50 > 10000 nM T20251 C6Z9PO 24951035 IC50 = 6000 nM T20251 CV0PG1 24951036 IC50 > 10000 nM T20251 CB03UR 24951038 IC50 = 5300 nM T20251 C02ADX 24951191 IC50 = 6700 nM T20251 C7WE9M 24951192 IC50 = 1600 nM T20251 CVT49O 24951193 IC50 > 10000 nM T20251 C7DGE0 24951348 IC50 = 2500 nM T20251 C9GA3W 24951349 IC50 = 2600 nM T20251 COW04Z 24951350 IC50 = 350 nM T20251 CHD86F 24951351 IC50 = 2800 nM T20251 CNP3T1 24951733 IC50 > 100000 nM T20251 C40XUR 24952765 IC50 = 30 nM T20251 CCO20I 24953169 Ki = 60 nM T20251 CC0U6X 24953170 Ki = 130 nM T20251 CO41IK 24953519 Ki = 180 nM T20251 C3AQG0 24957697 IC50 = 27500 nM T20251 C2JZ3S 24957698 IC50 > 30000 nM T20251 CZ3FO0 24958070 IC50 > 30000 nM T20251 C82OXU 24958071 IC50 > 30000 nM T20251 C6IC2O 24958072 IC50 > 30000 nM T20251 CB16FH 24958073 IC50 > 30000 nM T20251 C5H4QV 24958074 IC50 > 30000 nM T20251 CCJ9G0 24958075 IC50 > 30000 nM T20251 C04IDY 24958076 IC50 > 30000 nM T20251 C79TOJ 24958447 IC50 > 30000 nM T20251 CDTJ93 24958448 IC50 > 30000 nM T20251 CSF3J5 24958449 IC50 > 30000 nM T20251 CSZ1F5 24958450 IC50 > 30000 nM T20251 C9QX2O 24958451 IC50 > 30000 nM T20251 CAX05W 24958452 IC50 > 30000 nM T20251 CH4C3E 24958809 IC50 > 30000 nM T20251 CPC58S 24958810 IC50 > 30000 nM T20251 C14FUP 24958811 IC50 > 30000 nM T20251 CM94VS 24958812 IC50 > 30000 nM T20251 C65PZU 24958813 IC50 > 30000 nM T20251 C6YR5K 24958814 IC50 > 30000 nM T20251 CNX41V 24958815 IC50 > 30000 nM T20251 C2UZ5G 24958816 IC50 > 30000 nM T20251 C8BEW0 24959168 IC50 = 5200 nM T20251 CNO0U1 24959169 IC50 = 4800 nM T20251 C5J3SP 24959542 IC50 > 30000 nM T20251 CBM71O 24959543 IC50 = 22000 nM T20251 C5BZE7 24959906 IC50 = 2700 nM T20251 CC76EQ 24961017 IC50 = 14800 nM T20251 CR6C3N 24962469 IC50 = 3200 nM T20251 CW4X0E 24962988 Ki = 2830 nM T20251 C6EQG2 24963293 IC50 = 1790 nM T20251 C02YIQ 24963478 IC50 = 26000 nM T20251 CQ58IV 24964189 IC50 > 33000 nM T20251 CS6XP4 24964190 IC50 > 33000 nM T20251 CDC01R 24965775 IC50 = 54 nM T20251 CDF34R 24966125 IC50 = 320 nM T20251 CY0G1A 24966127 IC50 = 230 nM T20251 C6Z7KY 24967023 IC50 = 15000 nM T20251 C14KJT 24967024 IC50 > 33000 nM T20251 CY02UG 24967383 IC50 > 33000 nM T20251 CV40UK 24967750 IC50 > 32000 nM T20251 C4X1JN 24968454 IC50 = 22000 nM T20251 CYH04T 24968455 IC50 = 27000 nM T20251 C4D2VI 24968798 IC50 = 28000 nM T20251 CQ2Z7T 24985115 IC50 > 50118.72 nM T20251 CM7HQ5 24985395 IC50 > 200000 nM T20251 CEJ74C 24985745 IC50 > 200000 nM T20251 CNYD53 24987709 IC50 = 7900 nM T20251 CNMD47 24990839 IC50 = 2200 nM T20251 CZD3W7 24992427 IC50 = 380 nM T20251 CL83OS 24992519 IC50 > 10000 nM T20251 C16SVM 24992849 IC50 = 9000 nM T20251 C8KIP6 24993178 IC50 = 21000 nM T20251 CD8U2B 24993500 IC50 = 8000 nM T20251 CCDF20 24994127 IC50 > 10000 nM T20251 CK5LM1 24996644 IC50 = 7000 nM T20251 CFDQ56 24996645 IC50 > 30000 nM T20251 CTL2D0 24996647 IC50 = 2000 nM T20251 CPYC89 24998177 IC50 = 17000 nM T20251 C2DT4C 24998178 IC50 > 32000 nM T20251 CZ4OL9 24998808 IC50 = 8000 nM T20251 CVB1P5 24999737 IC50 > 32000 nM T20251 C21VCQ 25001553 IC50 = 11000 nM T20251 C6H4YL 25001554 IC50 = 14000 nM T20251 CUMH07 25001555 IC50 > 30000 nM T20251 CJR70I 25001557 IC50 > 30000 nM T20251 CIWR78 25001850 IC50 > 30000 nM T20251 CWO1V4 25004449 IC50 = 680 nM T20251 CETJ60 25006676 Ki = 19952.62 nM T20251 CN6J3R 25008249 IC50 = 93000 nM T20251 CYE9X4 25008593 IC50 = 176000 nM T20251 C5KNH1 25008765 IC50 = 305000 nM T20251 COE0T4 25008767 IC50 = 172000 nM T20251 CD2VF7 25008771 IC50 = 174000 nM T20251 C0KZ5Q 25008940 IC50 = 27000 nM T20251 CXB5T7 25008941 IC50 = 124000 nM T20251 CJ1HQ5 25009146 Ki = 10250 nM T20251 C7XMO2 25009310 Ki = 1760 nM T20251 CZ6T5Q 25009937 Ki = 3300 nM T20251 CCK8G4 25012362 IC50 = 1800 nM T20251 C0EI7T 25012524 IC50 = 277 nM T20251 C1VRJ3 25014630 IC50 = 13000 nM T20251 CM1H6K 25016328 IC50 > 10000 nM T20251 CV02TA 25017750 IC50 = 17000 nM T20251 CTYD20 25018000 IC50 = 11200 nM T20251 CJNR78 25018002 IC50 = 9100 nM T20251 C9AKD7 25018252 IC50 = 8400 nM T20251 CB36TF 25019018 IC50 = 26700 nM T20251 CUF48R 25019019 IC50 = 15800 nM T20251 C91QFN 25019282 IC50 = 15100 nM T20251 CKR94M 25022356 IC50 = 1000 nM T20251 CQ9LS6 25022704 Ki = 5800 nM T20251 C70MLG 25024304 IC50 = 81000 nM T20251 CA20NZ 25025581 IC50 = 4200 nM T20251 CNW89T 25026445 Ki = 4200 nM T20251 C5V1YO 25029711 IC50 = 4610 nM T20251 C8CIY2 25030810 IC50 > 30000 nM T20251 C6DO4B 25032525 Ki = 2202 nM T20251 C6K4SH 25033519 Ki > 7500 nM T20251 CVQS96 25052767 IC50 = 36000 nM T20251 CHQ86P 25054013 IC50 = 2300 nM T20251 C7EQ5T 25054288 IC50 = 9000 nM T20251 CCEY27 25054289 IC50 = 800 nM T20251 C0PIZ8 25054550 IC50 = 16000 nM T20251 C20JHU 25054551 IC50 > 30000 nM T20251 CG8C7J 25054804 IC50 = 2000 nM T20251 CJS39H 25055504 Ki = 5900 nM T20251 C1PKF0 25056080 IC50 > 10000 nM T20251 C0Z2SQ 25056787 IC50 = 10000 nM T20251 CPAZ91 25056788 IC50 = 7943.28 nM T20251 C2FP5D 25056872 IC50 = 16400 nM T20251 C6Z3CE 25057124 IC50 = 8500 nM T20251 C0TYE6 25057388 IC50 = 1800 nM T20251 CE12CD 25057645 IC50 > 30000 nM T20251 C1K9VQ 25057911 IC50 = 1800 nM T20251 CH4PI7 25057913 IC50 = 3300 nM T20251 C8L6JE 25058425 IC50 = 3 nM T20251 CR5FX4 25059765 IC50 = 0.65 nM T20251 CTI38U 25060119 IC50 = 6950 nM T20251 CMJ1F7 25067546 IC50 = 98000 nM T20251 C7YRG0 25067560 IC50 = 1584.89 nM T20251 CM83VQ 25067563 IC50 = 2800 nM T20251 C7O8YH 25068794 Ki = 779 nM T20251 CZ9SN8 25068797 Ki = 931 nM T20251 CL46IP 25068850 Ki = 1560 nM T20251 CEH7D9 25068903 Ki = 1680 nM T20251 CB03DL 25068905 Ki = 2810 nM T20251 C5ZHN9 25068906 Ki = 3610 nM T20251 C0ZJB7 25068907 Ki = 1290 nM T20251 C9G7EM 25068908 Ki = 439 nM T20251 C16ERI 25069015 Ki = 907 nM T20251 CHZB81 25069180 Ki = 1860 nM T20251 CBY3O2 25070582 IC50 > 22300 nM T20251 COE3T5 25071310 IC50 = 2511.89 nM T20251 CU0SR4 25071931 IC50 = 3981.07 nM T20251 C18XGM 25072242 IC50 = 1995.26 nM T20251 CG71VR 25072244 IC50 = 15848.93 nM T20251 C4RE0M 25072246 IC50 = 7943.28 nM T20251 CTWZ82 25072568 IC50 = 50118.72 nM T20251 CW2H9F 25072875 IC50 = 1995.26 nM T20251 CA4FV9 25072876 IC50 = 3981.07 nM T20251 CPUB18 25072877 IC50 = 1584.89 nM T20251 C6GPL3 25072880 IC50 = 794.33 nM T20251 CDY9Z4 25073188 IC50 = 12589.25 nM T20251 C3AJD0 25073189 IC50 = 6309.57 nM T20251 C9KR8V 25073190 IC50 = 10000 nM T20251 C68FHZ 25073191 IC50 = 2511.89 nM T20251 C98ISN 25073801 IC50 = 3981.07 nM T20251 C3AFU0 25093775 IC50 = 670 nM T20251 CP0IR1 25094630 IC50 > 32000 nM T20251 CKP3J6 25094902 IC50 > 25000 nM T20251 CNOA12 25094903 IC50 = 32000 nM T20251 CC6NZ8 25095678 IC50 > 33000 nM T20251 C2H4VG 25096016 IC50 = 1400 nM T20251 C51OJR 25099115 IC50 > 10000 nM T20251 CUB4W5 25102935 IC50 = 12000 nM T20251 CM0O7N 25102936 IC50 > 32000 nM T20251 C3PKV4 25102938 IC50 > 32000 nM T20251 CPM6S0 25104740 IC50 = 13000 nM T20251 CJW1T2 25104741 IC50 > 32000 nM T20251 C4S5XP 25107560 IC50 = 1390 nM T20251 CF1E3C 25107622 IC50 = 1910 nM T20251 CN7W1T 25107626 IC50 = 1630 nM T20251 C0BW7J 25107695 IC50 = 2400 nM T20251 C1XI8C 25107697 IC50 = 170 nM T20251 CUO18X 25107759 IC50 = 730 nM T20251 CC4YH9 25107761 IC50 = 830 nM T20251 CPL78K 25108016 IC50 = 370 nM T20251 C32VHJ 25108017 IC50 = 130 nM T20251 CN1B5F 25108078 IC50 = 430 nM T20251 COS8G5 25108135 IC50 = 1200 nM T20251 CGV7K5 25108137 IC50 = 1700 nM T20251 C5Q6GA 25108843 IC50 > 30000 nM T20251 CON1U6 25110598 IC50 = 12000 nM T20251 CQ2XF3 25110840 IC50 > 5000 nM T20251 CP03LT 25113806 IC50 = 2511.89 nM T20251 CWO19M 25114846 IC50 = 9970 nM T20251 CSI90H 25114847 IC50 = 85900 nM T20251 CDW2I9 25114850 IC50 = 7180 nM T20251 CS24RM 25115077 IC50 = 14100 nM T20251 C1D7TX 25115962 IC50 > 32000 nM T20251 CJC90O 25115964 IC50 > 32000 nM T20251 C2D9XW 25116186 IC50 = 52000 nM T20251 CMXE76 25116191 IC50 > 32000 nM T20251 C0QOD8 25117760 IC50 > 33000 nM T20251 CH57JF 25118124 IC50 > 33000 nM T20251 C6C0HA 25118125 IC50 > 33000 nM T20251 C4DMZ5 25118127 IC50 > 33000 nM T20251 CXBZ57 25118294 Ki = 400 nM T20251 CXE6T1 25118477 IC50 = 20800 nM T20251 CZ96TL 25118804 IC50 > 100000 nM T20251 C8T7NC 25118805 IC50 > 100000 nM T20251 CJM41E 25119356 Ki = 400 nM T20251 C8HI9Y 25119357 Ki = 500 nM T20251 CGL63Q 25119716 Ki = 500 nM T20251 CQ8Y7T 25120419 Ki = 1000 nM T20251 CS6O1Q 25120608 IC50 > 30000 nM T20251 C2G0BK 25120953 IC50 > 30000 nM T20251 CLV98T 25120954 IC50 > 30000 nM T20251 CXL3Q8 25121114 Ki = 600 nM T20251 C2S1LG 25121469 Ki = 200 nM T20251 CR2D3W 25122009 IC50 = 25000 nM T20251 C1RBQ7 25122183 Ki = 1070 nM T20251 CYWO57 25122184 Ki = 80 nM T20251 C07OMT 25122324 IC50 = 25000 nM T20251 C0KOU6 25123487 IC50 = 161 nM T20251 C0W8IC 25124143 IC50 = 1400 nM T20251 CL4XY0 25125138 IC50 = 100 nM T20251 CIYA24 25125139 IC50 = 720 nM T20251 CF54QZ 25129041 IC50 > 100000 nM T20251 CDO26T 25129042 IC50 = 7943.28 nM T20251 CUO63Q 25129091 IC50 = 379 nM T20251 CHK3S8 25129266 IC50 = 5000 nM T20251 CT9CL8 25129432 IC50 = 585 nM T20251 CLW14R 25129434 IC50 < 100 nM T20251 CQ36GH 25129435 IC50 = 663 nM T20251 C2XI7E 25129436 IC50 > 100000 nM T20251 CT30ZV 25129437 IC50 = 303 nM T20251 CM6KY3 25129438 IC50 = 6450 nM T20251 C5AF2Y 25129498 IC50 = 483 nM T20251 CDQ7C1 25129500 IC50 = 655 nM T20251 C5PA3S 25129777 IC50 = 47440 nM T20251 C9ELP5 25129778 IC50 = 1814 nM T20251 C5Q3JF 25129779 IC50 = 18310 nM T20251 C4DL2M 25129780 IC50 = 60000 nM T20251 CV93JO 25129849 IC50 = 2208 nM T20251 CL8YG2 25129850 IC50 = 883 nM T20251 CJ6TD3 25129852 IC50 = 1799 nM T20251 C8PJ6A 25129853 IC50 = 1047 nM T20251 C4SA9U 25129854 IC50 = 4823 nM T20251 C6CB1W 25130210 IC50 = 3674 nM T20251 CXK12T 25130211 IC50 = 1021 nM T20251 C6CF3U 25130212 IC50 = 2047 nM T20251 CS3OY1 25130213 IC50 = 4810 nM T20251 CGC5U6 25130214 IC50 = 4731 nM T20251 CYD2Q3 25130556 IC50 > 10000 nM T20251 CK04RW 25130557 IC50 = 1260 nM T20251 C3I1XJ 25132254 IC50 = 1995.26 nM T20251 C9J1MQ 25138078 IC50 = 24000 nM T20251 CC5O4P 25138090 IC50 = 540 nM T20251 CM03CP 25138344 IC50 > 50118.72 nM T20251 C9DQ8L 25139490 IC50 = 3900 nM T20251 CWL9E2 25139491 IC50 > 10000 nM T20251 C3XJM1 25139625 IC50 = 7300 nM T20251 CKLC61 25139757 IC50 = 5400 nM T20251 C4N1YF 25139758 IC50 = 3300 nM T20251 CFS3N9 25144422 IC50 = 860 nM T20251 CUX49Z 25144536 IC50 = 40900 nM T20251 C2H4KJ 25145553 IC50 = 740 nM T20251 CQR84M 25147644 IC50 = 54000 nM T20251 C35XQI 25150621 IC50 > 10000 nM T20251 CD0QU5 25150624 IC50 > 10000 nM T20251 CIZ1N9 25150625 IC50 > 10000 nM T20251 CE1ND3 25150628 IC50 > 10000 nM T20251 CAVR45 25150711 IC50 > 10000 nM T20251 CYOV03 25150901 IC50 > 30000 nM T20251 CMS9R3 25151607 IC50 > 30000 nM T20251 C0XBY4 25151662 IC50 > 30000 nM T20251 CD70KZ 25151793 IC50 = 2372 nM T20251 CHU1R7 25151849 IC50 > 30000 nM T20251 C7XDZ8 25151850 IC50 = 3580 nM T20251 CC1T8M 25151988 IC50 = 11330 nM T20251 CH9NA3 25151989 IC50 > 30000 nM T20251 C5AY6K 25151990 IC50 > 30000 nM T20251 CT3D7E 25152023 IC50 = 2310 nM T20251 C05HFO 25152653 IC50 > 30000 nM T20251 C8HXD1 25152860 IC50 > 30000 nM T20251 C7N4FW 25152862 IC50 > 30000 nM T20251 C68NWT 25153075 IC50 > 30000 nM T20251 CXC85P 25153077 IC50 = 1188 nM T20251 CZI56N 25153212 IC50 > 30000 nM T20251 CJW29T 25153282 IC50 = 12650 nM T20251 CR0EH4 25153700 IC50 > 30000 nM T20251 CH3M5P 25154041 IC50 = 3000 nM T20251 CI0E2L 25154395 IC50 = 2400 nM T20251 C4I1CJ 25155417 IC50 = 3000 nM T20251 CJVM09 25156194 Ki = 6600 nM T20251 C0TI3Z 25156476 Ki = 10000 nM T20251 CMX1W0 25156477 Ki = 220 nM T20251 C24UVQ 25156478 Ki = 870 nM T20251 C8AYP4 25156480 Ki = 620 nM T20251 C1HG2K 25156481 Ki = 2100 nM T20251 CKP4R2 25156482 Ki = 10000 nM T20251 CBM05I 25156750 Ki = 10000 nM T20251 C3QT7F 25156751 Ki = 10000 nM T20251 CJPO67 25156752 Ki = 10000 nM T20251 C7VC0P 25157642 IC50 > 5000 nM T20251 C7F1GA 25157660 IC50 = 3700 nM T20251 CP72MB 25159060 IC50 > 30000 nM T20251 CUAB05 25160153 IC50 = 1100 nM T20251 CGH08V 25164128 IC50 = 77.62 nM T20251 CW9MX8 25168440 IC50 > 10000 nM T20251 CYQ2X5 25170416 IC50 = 56 nM T20251 CZ28ES 25171661 IC50 > 32000 nM T20251 C5TJD2 25172265 IC50 > 30000 nM T20251 C94BLY 25173349 IC50 = 16000 nM T20251 C6AHF5 25174166 IC50 > 33000 nM T20251 CXG59Q 25175568 IC50 > 32000 nM T20251 C0YOQ7 25176461 IC50 = 9000 nM T20251 C1JL9X 25176462 IC50 = 5500 nM T20251 CL0Z1F 25181502 IC50 = 13000 nM T20251 C5C7GH 25184832 IC50 > 50118.72 nM T20251 C52BNH 25186023 Ki = 210 nM T20251 CJF9H4 25186569 Ki = 200 nM T20251 CG6NC3 25186839 Ki = 160 nM T20251 C3J8FK 25189510 IC50 = 95.5 nM T20251 CX4MV0 25190195 IC50 = 467.74 nM T20251 C1SX2E 25190435 IC50 = 630.96 nM T20251 CRS71Z 25190875 IC50 = 2700 nM T20251 C4AE8F 25190876 IC50 > 3000 nM T20251 CIR2T7 25190877 IC50 > 3000 nM T20251 C4XIE6 25190878 IC50 > 3000 nM T20251 CMZ83A 25190879 IC50 = 350 nM T20251 CG49HK 25190880 IC50 = 630 nM T20251 CHN5O0 25190977 IC50 = 10400 nM T20251 CV3TA6 25192021 IC50 > 3000 nM T20251 C7A8UE 25192471 IC50 > 3000 nM T20251 CH3L6V 25192656 IC50 > 30000 nM T20251 C6NA1J 25194889 IC50 = 178 nM T20251 C08QMV 25195086 Ki = 37.2 nM T20251 CD4L9N 25195087 Ki = 23.9 nM T20251 CNI57D 25195088 Ki > 100 nM T20251 CO8QV5 25195089 Ki > 100 nM T20251 CBK27L 25196164 IC50 > 30000 nM T20251 C19CNW 25196320 IC50 > 33000 nM T20251 C0MQ7R 25196433 IC50 > 33000 nM T20251 CHS15A 25196434 IC50 > 33000 nM T20251 C3F5HA 25196664 IC50 > 33000 nM T20251 CF2O6Z 25196665 IC50 > 33000 nM T20251 C58AOY 25196773 IC50 > 33000 nM T20251 CM5V0Q 25197117 IC50 > 31000 nM T20251 CF0O3T 25197227 IC50 > 33000 nM T20251 CT5P4U 25204216 IC50 = 700 nM T20251 CTQM87 25210756 IC50 > 100000 nM T20251 C2UQJ6 25211598 EC50 > 30000 nM T20251 CKI86X 25211805 EC50 > 30000 nM T20251 CHW2X0 25211910 EC50 > 30000 nM T20251 CK0AM3 25216601 IC50 > 30000 nM T20251 C3PZ7E 25216602 IC50 > 30000 nM T20251 CJ1Z9H 25216680 IC50 = 7400 nM T20251 C6EO8B 25216683 IC50 = 17000 nM T20251 CXK8C2 25217299 IC50 = 32500 nM T20251 CA8RO1 25217406 IC50 = 11300 nM T20251 CLHN01 25217407 IC50 = 8800 nM T20251 CT67WG 25217408 IC50 = 9300 nM T20251 CW7RJ2 25218015 IC50 = 300 nM T20251 CT3LJ6 25218017 IC50 = 140 nM T20251 C0VI2J 25218142 IC50 = 8800 nM T20251 C1T3LR 25218143 IC50 = 8200 nM T20251 C8RCG2 25218267 IC50 = 11000 nM T20251 C6VNQ4 25218268 IC50 = 16000 nM T20251 C0ONJ9 25218269 IC50 = 29000 nM T20251 CU63JR 25218271 IC50 = 6200 nM T20251 CPI03N 25218397 IC50 = 11000 nM T20251 C4GSU5 25218398 IC50 = 2500 nM T20251 CL1R3Q 25218401 IC50 = 9600 nM T20251 CN6XA4 25218555 IC50 = 1597 nM T20251 CL8K9U 25218556 IC50 = 1492 nM T20251 C9WA4B 25218557 IC50 = 183 nM T20251 CRG29Y 25218558 IC50 = 167 nM T20251 CEH71M 25218560 IC50 = 25090 nM T20251 C15YDI 25218563 IC50 = 12390 nM T20251 C9X6YJ 25229646 IC50 > 30000 nM T20251 CNF50T 25229676 Ki > 10000 nM T20251 C6FG0Q 25242540 IC50 > 30000 nM T20251 C53PTZ 25256089 IC50 > 10000 nM T20251 C90OGX 25256781 Ki = 5030 nM T20251 C2XS0Y 25256782 Ki = 903 nM T20251 CW9JM2 25256832 IC50 > 100000 nM T20251 C3GC7P 25256833 IC50 = 52000 nM T20251 C1IW5M 25261456 IC50 > 10000 nM T20251 CM81QH 25262336 IC50 > 32000 nM T20251 C20QHN 25262627 IC50 = 24200 nM T20251 C5E3ZH 25265089 IC50 = 37000 nM T20251 C20SGN 25265312 IC50 = 480 nM T20251 C5BNH3 25265516 IC50 = 18900 nM T20251 C7PK2X 29938807 IC50 > 33000 nM T20251 C60RHJ 30634189 IC50 = 320 nM T20251 CR6Q3D 34598448 IC50 = 24000 nM T20251 CJ8V4H 34681379 IC50 = 22900 nM T20251 C4GSR9 35901875 IC50 = 2238.72 nM T20251 CTI9S6 42601404 Ki = 2990 nM T20251 CQR2J6 42601405 Ki > 7200 nM T20251 CBQO98 42602095 IC50 = 7200 nM T20251 CJ61SE 42602096 IC50 = 6495 nM T20251 CI42XG 42602097 IC50 = 2600 nM T20251 CD2AH4 42602175 IC50 = 57793 nM T20251 CSWA85 42602176 IC50 > 100000 nM T20251 C1LUN4 42602178 IC50 > 100000 nM T20251 C8O3EA 42602260 IC50 > 100000 nM T20251 C93NKL 42602264 IC50 > 100000 nM T20251 C7WPJ5 42602351 IC50 > 33300 nM T20251 C2FZ9P 42606792 IC50 > 80000 nM T20251 CKH3P1 42606928 IC50 = 1900 nM T20251 CIH75Y 42615261 IC50 > 30000 nM T20251 C1YO7H 42618040 EC50 = 12000 nM T20251 CGU3N8 42618068 EC50 = 8000 nM T20251 CY4LG8 42622934 IC50 = 22000 nM T20251 CI1C5U 42623163 IC50 = 4000 nM T20251 CV3FM2 42625548 IC50 = 900 nM T20251 CZ96KC 42625549 IC50 = 2500 nM T20251 C1U5IS 42625550 IC50 = 60 nM T20251 C9GPZ5 42625636 IC50 = 500 nM T20251 C4C5QJ 42625708 IC50 = 1300 nM T20251 C5XVB9 42625945 IC50 = 1200 nM T20251 CZ4V2A 42625948 IC50 = 1200 nM T20251 C2VA7M 42625949 IC50 = 500 nM T20251 CQ1YN9 42626020 IC50 = 40 nM T20251 C7K6PG 42626023 IC50 = 3500 nM T20251 CJ8LY0 42626024 IC50 = 1000 nM T20251 CRQ91B 42626318 IC50 = 380 nM T20251 CNU7P4 42630820 IC50 > 10000 nM T20251 C1CWU0 42631007 IC50 = 6850 nM T20251 CW24IK 42633780 IC50 = 700 nM T20251 C75GFD 42633960 IC50 > 10000 nM T20251 C57VJY 42635854 IC50 = 3400 nM T20251 CP8RA7 42635855 IC50 = 3000 nM T20251 CG0E4V 42635876 IC50 = 17782.79 nM T20251 C05BWT 42635901 IC50 = 8200 nM T20251 CY5E4B 42635983 IC50 = 1700 nM T20251 C8V6IK 42635984 IC50 = 990 nM T20251 C34DCR 42636018 IC50 = 750 nM T20251 C1J4XZ 42636222 IC50 > 30000 nM T20251 C9PL8Z 42641334 Ki = 5000 nM T20251 C6MX0U 42641453 IC50 = 4500 nM T20251 CZM36T 42641892 IC50 = 1400 nM T20251 CA5TW1 42641905 Ki = 2200 nM T20251 CQS4U7 42642010 Ki = 680 nM T20251 CIX54O 42642011 Ki = 1000 nM T20251 CRYH80 42642459 IC50 = 2700 nM T20251 CZF5G9 42916879 IC50 > 50000 nM T20251 C0VC7J 43314210 IC50 = 20000 nM T20251 CYV94L 43314375 IC50 = 4560 nM T20251 CXYI49 44121506 IC50 > 33000 nM T20251 CS40ML 44123747 IC50 = 30000 nM T20251 CD61KH 44125830 IC50 = 95499.26 nM T20251 CPB8S3 44125832 IC50 = 18197.01 nM T20251 C1BT4A 44129293 IC50 = 3162.28 nM T20251 C1HZK2 44135978 IC50 = 3300 nM T20251 C1HRC7 44135979 IC50 = 3300 nM T20251 CA7HI4 44137226 IC50 = 2100 nM T20251 CSX10M 44138030 IC50 = 18000 nM T20251 CXZH39 44138098 Ki = 2511.89 nM T20251 CG73ST 44138103 IC50 > 30000 nM T20251 CUOD42 44138104 Ki = 3981.07 nM T20251 CSM1A0 44138577 IC50 = 490 nM T20251 C4VYG8 44138579 IC50 > 10000 nM T20251 C3WOD7 44138581 IC50 > 10000 nM T20251 C4P8OL 44138706 IC50 > 10000 nM T20251 CW2G7S 44138708 IC50 = 7800 nM T20251 C7H3NP 44138709 IC50 > 10000 nM T20251 CU4XB0 44139234 IC50 = 1730 nM T20251 CDF14X 44139355 IC50 = 490 nM T20251 C4Q9IL 44139356 IC50 > 10000 nM T20251 CG3KU0 44139478 IC50 > 10000 nM T20251 CXR3J2 44139479 IC50 = 4330 nM T20251 CW8J0K 44139480 IC50 > 10000 nM T20251 COJK15 44139481 IC50 = 6930 nM T20251 CX17RC 44139599 IC50 = 6330 nM T20251 CY0GQ3 44139600 IC50 > 10000 nM T20251 CVCH41 44139601 IC50 > 10000 nM T20251 C79OCX 44139602 IC50 > 10000 nM T20251 C9Z0RV 44139603 IC50 > 10000 nM T20251 C2U9ES 44139732 IC50 = 6300 nM T20251 C49YRK 44143406 IC50 = 23 nM T20251 C6U7HP 44143413 IC50 = 23 nM T20251 CAB3T9 44143415 IC50 = 2900 nM T20251 CG3PW7 44143417 IC50 = 23000 nM T20251 CB94OV 44143418 IC50 = 2700 nM T20251 COP5W8 44143419 IC50 = 16000 nM T20251 C3S1PL 44143422 IC50 = 9000 nM T20251 CQE5U4 44143426 IC50 = 1200 nM T20251 CZR49E 44143427 IC50 = 30000 nM T20251 C63RXB 44143428 IC50 = 29000 nM T20251 C8OH4S 44143429 IC50 = 21000 nM T20251 CTE6S1 44143430 IC50 = 23000 nM T20251 CL57VS 44143431 IC50 = 41000 nM T20251 C2C5QW 44143432 IC50 = 1500 nM T20251 C6GDL8 44143433 IC50 > 10000 nM T20251 C3BNV0 44143434 IC50 = 4900 nM T20251 CXV0B8 44143435 IC50 = 3000 nM T20251 CN7HE0 44143436 IC50 = 8500 nM T20251 C9CJN0 44143437 IC50 = 11000 nM T20251 C6INT4 44143438 IC50 = 990 nM T20251 CJ46YA 44143439 IC50 > 10000 nM T20251 C0KB7Y 44143441 IC50 > 10000 nM T20251 C3RF4I 44143442 IC50 > 10000 nM T20251 C5NZM3 44143446 IC50 = 3900 nM T20251 CGSW03 44143448 IC50 > 10000 nM T20251 CBWD06 44143449 IC50 > 10000 nM T20251 C2ST5N 44143450 IC50 > 10000 nM T20251 CF4V5K 44143451 IC50 > 10000 nM T20251 CL3R6D 44143452 IC50 > 10000 nM T20251 C8IG1V 44143453 IC50 = 4400 nM T20251 C2Q3DE 44143454 IC50 = 6300 nM T20251 CZX75A 44143455 IC50 = 380 nM T20251 C02YJQ 44143456 IC50 = 3400 nM T20251 CZV0C7 44143457 IC50 > 10000 nM T20251 C6TND7 44155109 IC50 = 8400 nM T20251 CN5G6U 44156749 IC50 = 100 nM T20251 C2C4NJ 44156750 IC50 = 7400 nM T20251 C6UOJ1 44157408 IC50 > 10000 nM T20251 CAS7T0 44157572 IC50 > 10000 nM T20251 CHI65U 44159530 IC50 > 30000 nM T20251 CE3OF9 44160137 IC50 = 750 nM T20251 CU2PO5 44180522 IC50 = 25118.86 nM T20251 CPF50A 44184875 IC50 = 17000 nM T20251 C2XE7Y 44189733 IC50 = 25000 nM T20251 C1ML3E 44190627 IC50 > 10000 nM T20251 C2AV1K 44190762 IC50 = 3230 nM T20251 CP06EY 44199337 IC50 = 28000 nM T20251 CJ7AF4 44203948 IC50 = 5000 nM T20251 CMR7T1 44204999 IC50 = 79.43 nM T20251 C4TMP9 44205087 IC50 > 30000 nM T20251 CX54AP 44215433 IC50 = 4400 nM T20251 CT29ZS 44216196 Ki = 2702 nM T20251 C2KJB0 44216880 IC50 = 1400 nM T20251 CUQ4T9 44217080 EC50 = 7943.28 nM T20251 CCJ3S4 44222256 Ki = 4650 nM T20251 CE0U8G 44222257 Ki = 7900 nM T20251 CC3XR6 44222258 Ki = 22500 nM T20251 CRNL71 44225654 Ki = 2900 nM T20251 C3MR8P 44229544 IC50 > 10000 nM T20251 CGPI02 44229545 IC50 > 10000 nM T20251 C83NXZ 44229546 IC50 > 10000 nM T20251 CQ4TG8 44229547 IC50 = 8300 nM T20251 CUVJ20 44229621 IC50 = 1600 nM T20251 CB5P7N 44230873 IC50 > 30000 nM T20251 CIBR82 44231149 IC50 > 10000 nM T20251 CX4YL8 44232522 IC50 > 30000 nM T20251 CMKQ59 44233027 IC50 = 19400 nM T20251 CQ13MH 44234032 IC50 > 30000 nM T20251 C7UY5F 44235863 IC50 > 30000 nM T20251 CX2W8Y 44236320 IC50 = 8000 nM T20251 C8LN0U 44236321 IC50 = 25000 nM T20251 CK4S5Y 44236322 IC50 = 6000 nM T20251 C75UQR 44236568 IC50 > 25000 nM T20251 CK7F2E 44240743 IC50 = 1300 nM T20251 C4W0SH 44247585 IC50 = 3200 nM T20251 C7MY2N 44247806 IC50 = 1400 nM T20251 CF9TE1 44247935 IC50 = 1200 nM T20251 CJ8RW5 44249745 IC50 = 7943.28 nM T20251 CLX51J 44249749 IC50 = 50118.72 nM T20251 C7QS6G 44250210 IC50 = 11400 nM T20251 C64ASH 44250211 IC50 = 26600 nM T20251 C85DHY 44250284 Ki = 18 nM T20251 C8P2LE 44250288 IC50 = 4900 nM T20251 C2K0VZ 44253016 IC50 > 63095.73 nM T20251 CY0QB9 44253226 IC50 = 3810 nM T20251 C1O8LH 44253973 IC50 = 12653 nM T20251 CMD87L 44254048 IC50 = 7000 nM T20251 C47RZO 44254057 IC50 = 2543 nM T20251 C41MNG 44254058 IC50 = 1261 nM T20251 C2SVL6 44254059 IC50 = 5132 nM T20251 CVW13I 44254060 IC50 = 3463 nM T20251 C0NZW8 44254061 IC50 = 71666 nM T20251 C3N2KB 44254062 IC50 = 4485 nM T20251 CJW3P2 44254063 IC50 = 4243 nM T20251 CXA10D 44254307 IC50 = 1918.03 nM T20251 C6OJS0 44254504 IC50 = 3190 nM T20251 CSBD48 44254505 IC50 = 23070 nM T20251 C1IPQ6 44254506 IC50 = 10566 nM T20251 CTL57U 44254584 IC50 = 54256 nM T20251 CZY2S1 44254585 IC50 = 1571 nM T20251 C9SQ8D 44254859 IC50 > 100000 nM T20251 CB47EJ 44254954 IC50 = 6809 nM T20251 C79QBX 44254955 IC50 = 3027 nM T20251 CVCP62 44254956 IC50 = 3501 nM T20251 CK7B1Q 44254957 IC50 = 13500 nM T20251 CJH6K5 44255041 IC50 = 6429 nM T20251 C5Z9KH 44255042 IC50 = 18471 nM T20251 C1FE8D 44255043 IC50 > 100000 nM T20251 CGB3A7 44255044 IC50 = 3794 nM T20251 CTY9U6 44255045 IC50 = 418 nM T20251 CZXC86 44267871 IC50 = 4360 nM T20251 CLC2O3 44294224 Ki = 1200 nM T20251 CO37IY 44294481 Ki = 1900 nM T20251 CV80DA 44294519 Ki = 400 nM T20251 C37OCJ 44294535 Ki = 460 nM T20251 CLHM64 44294659 Ki = 2200 nM T20251 CK7E2B 44294660 Ki = 490 nM T20251 CR2W3U 44294689 Ki = 1400 nM T20251 CCB5Y4 44296949 IC50 = 457.09 nM T20251 CE1S8X 44297083 IC50 = 36.31 nM T20251 CDSI60 44297084 IC50 = 10000 nM T20251 CE9H3D 44297095 IC50 = 2200 nM T20251 CP0T8C 44297148 IC50 = 10000 nM T20251 CD74SU 44297164 IC50 = 26000 nM T20251 CG9E7X 44297171 IC50 = 23.44 nM T20251 CR92VP 44297212 IC50 = 10000 nM T20251 CSX1R4 44297356 IC50 = 1947 nM T20251 C1VF2S 44297363 IC50 = 15848.93 nM T20251 C71ZUL 44297364 IC50 = 4570881.9 nM T20251 C96MUT 44297365 IC50 = 1480 nM T20251 C4MRW5 44297377 IC50 = 75000 nM T20251 C2FSL4 44297378 IC50 = 131 nM T20251 C5ZYX2 44297395 IC50 = 575.44 nM T20251 C3PX0Q 44297409 IC50 = 137 nM T20251 C0LT3N 44297410 IC50 = 87.1 nM T20251 C09HMY 44305854 Ki = 600 nM T20251 CMIB37 44306212 Ki > 10000 nM T20251 C70XSQ 44317802 Ki = 42200 nM T20251 C9AV2P 44326600 IC50 = 5888.44 nM T20251 CKSO92 44360724 Ki > 100000 nM T20251 CYED53 44360725 Ki = 5700 nM T20251 C50NME 44360749 Ki = 40000 nM T20251 CXTP74 44360787 Ki > 100000 nM T20251 C5MB1D 44360809 Ki = 17000 nM T20251 C29DTA 44360810 Ki = 29000 nM T20251 CR7Q9N 44360911 Ki = 5900 nM T20251 C6IZ8L 44360955 Ki = 22000 nM T20251 CY8A9K 44361010 Ki = 1900 nM T20251 CMU02Q 44364616 Ki = 20 nM T20251 C1XOB5 44387732 Ki = 1525 nM T20251 CL54KN 44387733 Ki = 398 nM T20251 C80WKC 44387740 Ki = 6800 nM T20251 CROA61 44387743 Ki = 9971 nM T20251 C1M5OY 44387746 Ki = 2446 nM T20251 CK36VZ 44387776 Ki > 9000 nM T20251 CC0WK5 44387777 Ki > 9000 nM T20251 CQ9WS8 44387780 Ki = 397 nM T20251 CY09ES 44396504 IC50 > 30000 nM T20251 C4X2OS 44396541 IC50 = 76800 nM T20251 CY80RP 44396542 IC50 = 800 nM T20251 C16MBG 44401760 IC50 < 10000 nM T20251 CC4O3R 44402387 IC50 = 180 nM T20251 C08LKH 44402452 IC50 = 30 nM T20251 CFA9P3 44402564 IC50 = 151.36 nM T20251 CXJ0Z6 44402597 IC50 = 40 nM T20251 CZI0A4 44405840 IC50 = 3.2 nM T20251 CH7Z3D 44407321 Ki = 4800 nM T20251 CFU2S7 44407325 Ki = 240 nM T20251 CE2R3O 44407331 Ki = 420 nM T20251 CHO57T 44407370 Ki = 190 nM T20251 CS21QZ 44407422 Ki > 5000 nM T20251 CLG2U0 44407427 Ki = 360 nM T20251 CUTS73 44407431 Ki > 6000 nM T20251 CCQX09 44407459 Ki > 6000 nM T20251 C9B4AK 44407467 Ki = 1400 nM T20251 CDPQ01 44407513 Ki = 270 nM T20251 CRB41P 44408123 Ki = 798 nM T20251 CQPK26 44408124 Ki = 1996 nM T20251 C92YHJ 44408144 Ki = 984 nM T20251 C35UHG 44408158 Ki = 3706 nM T20251 CF05TZ 44408176 Ki = 327 nM T20251 CA94TU 44408177 Ki = 947 nM T20251 CK4IB0 44408290 Ki = 1946 nM T20251 CDK7W3 44408291 Ki = 2987 nM T20251 CTM53U 44408295 Ki = 6529 nM T20251 CJE43Y 44408313 Ki = 862 nM T20251 COH25L 44409031 IC50 = 40000 nM T20251 CWX62Y 44409096 IC50 = 21000 nM T20251 CG87PW 44409290 IC50 > 30000 nM T20251 CB91NT 44409718 IC50 = 7800 nM T20251 C5YP1R 44409879 IC50 = 7800 nM T20251 CKI20Y 44409884 IC50 = 15000 nM T20251 C39MWE 44409885 IC50 = 6600 nM T20251 CF8A0Z 44409903 IC50 = 8500 nM T20251 CYO7B5 44409904 IC50 = 5600 nM T20251 C7BM2G 44409905 IC50 = 18000 nM T20251 CP10EK 44410155 Ki = 1300 nM T20251 C3YC0E 44410191 Ki = 1930 nM T20251 C5I4SO 44410193 Ki = 100 nM T20251 CY69JU 44410194 Ki = 1250 nM T20251 C5QG1S 44410207 Ki = 3150 nM T20251 CVB31D 44410278 Ki = 1800 nM T20251 CKWZ76 44410281 Ki = 2800 nM T20251 CQ8T0X 44410283 Ki > 10000 nM T20251 CYT96G 44410317 Ki > 5000 nM T20251 CYP37K 44410821 Ki = 150 nM T20251 CJI8T3 44410823 Ki = 150 nM T20251 C01JXU 44410838 Ki = 160 nM T20251 C1LYC9 44410849 Ki = 88 nM T20251 CGF17I 44410876 Ki = 135 nM T20251 CF0O7N 44410878 Ki = 1800 nM T20251 CL1XV7 44410904 Ki = 310 nM T20251 C4P5TW 44410944 Ki > 2000 nM T20251 CAO78Q 44411663 Ki > 9000 nM T20251 C8NVH0 44411664 Ki > 9000 nM T20251 C2Y8VK 44411667 Ki > 9000 nM T20251 C38VWG 44411668 Ki = 4869 nM T20251 C5Z2IY 44411674 Ki > 9000 nM T20251 CU2EY5 44411847 Ki > 9000 nM T20251 CD0OH1 44411864 Ki > 9000 nM T20251 CTLN43 44411929 Ki > 9000 nM T20251 CKX6D2 44411930 Ki > 9000 nM T20251 CQ89KF 44411933 Ki > 9000 nM T20251 CCJ1S9 44411934 Ki > 9000 nM T20251 CL28ZA 44411935 Ki > 9000 nM T20251 CG13DQ 44411936 Ki > 9000 nM T20251 CUB0V6 44412159 Ki > 9000 nM T20251 CO82EW 44412173 Ki = 1800 nM T20251 CACE19 44412207 Ki > 9000 nM T20251 CV4KZ7 44412225 Ki > 9000 nM T20251 CHF80Z 44412226 Ki > 9000 nM T20251 CCD01F 44412235 Ki = 1400 nM T20251 CECW41 44412236 Ki > 9000 nM T20251 C1D7YV 44412245 Ki > 9000 nM T20251 CH04GP 44412373 Ki = 5400 nM T20251 CYK1I6 44412374 Ki = 6700 nM T20251 CK5O6Q 44412445 Ki = 2400 nM T20251 CW71MS 44412453 Ki > 9000 nM T20251 C6R2ID 44412493 Ki = 8500 nM T20251 CDT7U5 44414663 IC50 > 24000000 nM T20251 CQD2S5 44414696 IC50 = 10900 nM T20251 C5Y4NH 44415354 IC50 = 170 nM T20251 C0OG4J 44415524 IC50 = 2600 nM T20251 CG1WM8 44417887 IC50 = 3300 nM T20251 CK76AM 44417889 IC50 = 3300 nM T20251 CPE50S 44417890 IC50 = 5860 nM T20251 CQS6G2 44417891 IC50 = 1700 nM T20251 CAK9U7 44417893 IC50 = 4000 nM T20251 C35KLS 44417895 IC50 = 5000 nM T20251 CL5XO4 44417897 IC50 = 25000 nM T20251 CM9QI8 44417899 IC50 = 14600 nM T20251 CI16UJ 44417902 IC50 = 26700 nM T20251 C8GK5Q 44417904 IC50 = 1800 nM T20251 C9BDI1 44417906 IC50 = 20000 nM T20251 C3GW2E 44417908 IC50 = 24000 nM T20251 CN2G7U 44417910 IC50 = 25000 nM T20251 CPDW02 44417913 IC50 = 10000 nM T20251 CY46AB 44417914 IC50 = 25000 nM T20251 C5HA7X 44417916 IC50 = 14000 nM T20251 CW1D3V 44417919 IC50 = 2600 nM T20251 C3CM4J 44417922 IC50 = 5100 nM T20251 CH0T1F 44417923 IC50 = 11000 nM T20251 C4WU0N 44417924 IC50 = 13000 nM T20251 CE96RJ 44417926 IC50 = 5200 nM T20251 C27PHW 44417927 IC50 = 13200 nM T20251 CT0B1U 44417929 IC50 = 2000 nM T20251 CH08OA 44417936 IC50 = 85200 nM T20251 CH3QM1 44417938 IC50 = 60700 nM T20251 CP1U0Z 44417939 IC50 = 5790 nM T20251 C7CP8I 44417993 IC50 = 20000 nM T20251 C6Q7ZM 44418004 IC50 = 6700 nM T20251 CVF74L 44418464 IC50 = 5151.52 nM T20251 C04THX 44418471 IC50 = 28461.54 nM T20251 CS6PZ7 44418472 IC50 = 19411.76 nM T20251 C9XDL2 44418473 IC50 = 52500 nM T20251 C49MQF 44418477 IC50 = 12222.22 nM T20251 CQ2D0O 44418482 IC50 = 101111.11 nM T20251 CPTD84 44418489 IC50 = 37619.05 nM T20251 CX09NV 44418490 IC50 = 66923.08 nM T20251 C68QUP 44418491 IC50 = 115000 nM T20251 CV5PD9 44418497 IC50 = 115000 nM T20251 CU8B2E 44418498 IC50 = 52500 nM T20251 C6YX3F 44418499 IC50 = 22258.06 nM T20251 CUH08F 44418511 IC50 = 40000 nM T20251 CR9EN2 44418522 Ki = 5100 nM T20251 C2S4RW 44418978 Ki = 1800 nM T20251 C93VJL 44418979 Ki = 6500 nM T20251 C16FUK 44418980 Ki = 510 nM T20251 CS08LV 44418981 Ki = 530 nM T20251 CP9VN3 44418982 Ki = 2500 nM T20251 CS5EY1 44418983 Ki = 8000 nM T20251 CHF36T 44418984 Ki = 2000 nM T20251 CF1A6T 44418985 Ki > 9000 nM T20251 C85GLF 44418986 Ki > 9000 nM T20251 CHS73F 44418998 Ki = 3000 nM T20251 C1FM8H 44419014 Ki = 8900 nM T20251 C5MT2W 44419015 Ki = 880 nM T20251 C7GY8W 44419017 Ki = 520 nM T20251 CW1DP9 44419019 Ki = 8200 nM T20251 C9H0DC 44419033 Ki > 9000 nM T20251 CT9U3N 44419048 Ki = 370 nM T20251 CR4SW2 44419049 Ki = 51 nM T20251 CP92ZY 44419050 Ki = 600 nM T20251 CO78NZ 44419051 Ki > 10000 nM T20251 CP85IH 44419052 Ki > 10000 nM T20251 C7OI8A 44419059 Ki = 4900 nM T20251 CCY70M 44419061 Ki = 840 nM T20251 C8PJ6U 44419062 Ki = 320 nM T20251 CCIF05 44419082 Ki = 71 nM T20251 CZNH91 44419083 Ki = 17 nM T20251 CRM0E4 44419084 Ki > 10000 nM T20251 CUI95V 44419085 Ki > 10000 nM T20251 C9LPR4 44419087 Ki > 10000 nM T20251 CQR29N 44419088 Ki = 880 nM T20251 CSQ5G8 44419089 Ki > 10000 nM T20251 COJ27C 44419090 Ki = 1400 nM T20251 CJ0W7B 44419091 Ki = 1400 nM T20251 C8LV0Y 44419092 Ki = 140 nM T20251 CDN8K7 44419097 Ki > 2000 nM T20251 C1A0LP 44419098 Ki = 1000 nM T20251 C3LE0S 44419101 Ki = 1600 nM T20251 C1VCN7 44419103 Ki = 89 nM T20251 CQ7PD9 44419104 Ki > 10000 nM T20251 C06ELF 44419105 Ki = 71 nM T20251 C7XKO9 44419106 Ki > 6600 nM T20251 CPL39F 44419108 Ki = 4600 nM T20251 CID32E 44419109 Ki = 200 nM T20251 C7HDX0 44419112 Ki = 570 nM T20251 C54KZH 44419113 Ki > 10000 nM T20251 C0J4HZ 44419117 Ki > 10000 nM T20251 CX5NU8 44419120 Ki = 790 nM T20251 CSIJ84 44419121 Ki > 10000 nM T20251 COV56X 44419122 Ki > 10000 nM T20251 CXZ2L3 44421702 IC50 = 5360 nM T20251 CT0J7Z 44421703 IC50 = 1410 nM T20251 CT03MH 44424972 Ki = 3.6 nM T20251 CEA35L 44424973 Ki = 7300 nM T20251 C3U2GQ 44424974 Ki = 160 nM T20251 CRV85N 44424975 Ki = 18 nM T20251 C4IRD2 44424976 Ki = 13 nM T20251 C7HW6E 44424977 Ki = 7 nM T20251 CDXQ90 44424979 Ki = 19 nM T20251 CXS4T5 44424981 Ki = 10 nM T20251 CIH6L7 44424983 Ki = 15 nM T20251 C53YCH 44424984 Ki = 89 nM T20251 C42IGZ 44424985 Ki > 1000 nM T20251 C6JW9A 44425428 Ki = 24000 nM T20251 CU43XH 44425429 Ki = 106000 nM T20251 C1JS6T 44425430 Ki > 150000 nM T20251 C2OSP1 44425431 Ki > 150000 nM T20251 CSR6M2 44425432 Ki = 64000 nM T20251 C02HMN 44425433 Ki > 100000 nM T20251 CUWC08 44425434 Ki > 100000 nM T20251 CZ7IT9 44425435 Ki > 150000 nM T20251 CI94RJ 44425436 Ki = 72000 nM T20251 CH6B9Z 44425437 Ki > 100000 nM T20251 C5Y6CS 44425438 Ki > 150000 nM T20251 C8OR0K 44425439 Ki > 150000 nM T20251 C56HGJ 44425440 Ki = 112000 nM T20251 CL0DM4 44425441 Ki > 150000 nM T20251 C53ELI 44425442 Ki = 45000 nM T20251 CCRH08 44428207 IC50 = 251.19 nM T20251 CTD5N2 44430312 IC50 > 30000 nM T20251 CON04H 44430571 IC50 = 7100 nM T20251 CCBR69 44430578 IC50 = 15900 nM T20251 C9GIE3 44433617 IC50 > 100000 nM T20251 C6VLC5 44433700 IC50 > 30000 nM T20251 CM0FX1 44433701 IC50 > 30000 nM T20251 CN24TK 44433702 IC50 > 10000 nM T20251 C1QH9B 44433704 IC50 > 30000 nM T20251 CWL6Z1 44433706 IC50 > 30000 nM T20251 C3CS8V 44433710 IC50 > 30000 nM T20251 C6UVW9 44433711 IC50 > 30000 nM T20251 CKVG69 44433749 IC50 > 30000 nM T20251 CEX75D 44435377 IC50 = 15900 nM T20251 CJ1ST3 44437610 Ki = 56 nM T20251 CY9IK3 44438461 Ki = 98.1 nM T20251 C6W2EZ 44438462 Ki = 261 nM T20251 C9IFR5 44438464 Ki = 205 nM T20251 CUB30F 44438465 Ki = 693 nM T20251 CE36YV 44438467 Ki = 709 nM T20251 CLWE65 44438469 Ki = 525 nM T20251 CI93VE 44438472 Ki = 1300 nM T20251 CXD9B1 44438473 Ki = 410 nM T20251 C0QEB9 44438474 Ki = 222 nM T20251 C9T7JL 44438740 IC50 = 65000 nM T20251 CB9S3W 44438741 IC50 = 4300 nM T20251 CL20OD 44438742 IC50 = 1600 nM T20251 CG3PZ7 44438744 IC50 = 34000 nM T20251 C71UWM 44438745 IC50 = 740 nM T20251 CBJ5R9 44438747 IC50 = 3200 nM T20251 C5VFD8 44438748 IC50 = 450 nM T20251 CW8GU6 44438753 IC50 = 6300 nM T20251 CS9D3H 44438755 IC50 = 6600 nM T20251 CQ18PR 44439374 Ki > 9000 nM T20251 CN9RH5 44439375 Ki > 9000 nM T20251 C2X1FS 44439377 Ki > 9000 nM T20251 CW2KQ1 44439378 Ki = 4200 nM T20251 C2J9LG 44439379 Ki = 4800 nM T20251 COKH57 44439380 Ki = 5000 nM T20251 CO20GU 44439381 Ki = 1500 nM T20251 C4KQ8C 44439384 Ki = 1400 nM T20251 CQXS03 44439385 Ki = 2900 nM T20251 C1R0DN 44441341 Ki > 7500 nM T20251 C2GAV7 44441348 IC50 = 2900 nM T20251 C61VKY 44441350 IC50 = 1600 nM T20251 CF4A8D 44441351 IC50 = 2400 nM T20251 CD30KT 44441353 IC50 = 1200 nM T20251 CG5KW9 44442083 IC50 > 30000 nM T20251 COX3Q2 44442283 IC50 = 3300 nM T20251 C2X7NQ 44442481 IC50 = 2600 nM T20251 CAC7V9 44442482 IC50 = 2400 nM T20251 CVO5Z2 44442483 IC50 = 1600 nM T20251 CJPR25 44442484 IC50 = 7400 nM T20251 C9NMQ3 44442485 IC50 = 3100 nM T20251 CLX76D 44442486 IC50 = 16000 nM T20251 CZF32M 44442487 IC50 = 3300 nM T20251 C8S9AX 44442488 IC50 = 10000 nM T20251 C01RSY 44442489 IC50 < 1500 nM T20251 CGM63L 44442490 IC50 < 1000 nM T20251 C83FXU 44442491 IC50 = 11000 nM T20251 C52VPZ 44443347 IC50 = 1800 nM T20251 C7M0HV 44443354 IC50 = 165000 nM T20251 CUG6X5 44443360 IC50 = 10000 nM T20251 CP7WL5 44443363 IC50 = 28900 nM T20251 CPN7J9 44443420 IC50 > 300000 nM T20251 CXQP15 44443798 IC50 = 5300 nM T20251 CUHO63 44443803 IC50 = 13200 nM T20251 CIH69B 44445848 IC50 = 800 nM T20251 C5RVE0 44446999 Ki = 101 nM T20251 C9E0FL 44447001 Ki = 616 nM T20251 CSJ4U5 44447002 Ki = 164 nM T20251 CL87PU 44447003 Ki = 196 nM T20251 CCD6B5 44447005 Ki = 35 nM T20251 CBH65G 44447007 Ki = 278 nM T20251 C8CF7X 44447008 Ki = 272 nM T20251 CN3EH7 44447010 Ki = 194 nM T20251 CYWP06 44447012 Ki = 166 nM T20251 C41KNM 44447013 Ki = 78 nM T20251 CE12BC 44447015 Ki = 358 nM T20251 CUD31L 44447018 Ki = 201 nM T20251 CNLX79 44447028 Ki = 511 nM T20251 CM8K1H 44447039 Ki = 35 nM T20251 C5IJW2 44447059 Ki = 150 nM T20251 CHXF10 44447061 Ki = 143 nM T20251 CG93OH 44447063 Ki = 184 nM T20251 C9KJR2 44447065 Ki = 269 nM T20251 C5QK8Z 44447067 Ki = 137 nM T20251 C7A6RP 44447068 Ki = 219 nM T20251 CM8P9A 44447070 Ki = 135 nM T20251 CK4HA6 44447072 Ki = 202 nM T20251 C9EM8Q 44447733 IC50 = 410 nM T20251 CX89DC 44447734 IC50 = 2000 nM T20251 CI8Q9M 44447766 IC50 = 16 nM T20251 C50JFH 44447775 IC50 = 45 nM T20251 CWY54R 44447782 IC50 = 217 nM T20251 C2UGM9 44447783 IC50 = 67 nM T20251 CSLU08 44447786 IC50 = 2786 nM T20251 CRV6F7 44447789 IC50 = 19720 nM T20251 CDI1F4 44447815 IC50 = 186 nM T20251 C5K8ZM 44447866 IC50 > 100000 nM T20251 C8W5YG 44447872 IC50 > 100000 nM T20251 CRO52K 44448053 Ki = 180 nM T20251 CJC38Z 44449333 Ki > 7500 nM T20251 COP8A3 44449880 IC50 = 5610 nM T20251 CGR0B6 44452775 IC50 > 20000 nM T20251 CDS52W 44453970 IC50 = 47000 nM T20251 CB1MX2 44454118 IC50 = 6309.57 nM T20251 CR3IC6 44454120 IC50 = 31622.78 nM T20251 C5B0IF 44454150 IC50 = 1584.89 nM T20251 CRD82N 44454166 IC50 = 3981.07 nM T20251 CMVS90 44454167 IC50 > 15848.93 nM T20251 C7FY1E 44454168 IC50 = 6309.57 nM T20251 CW4S3P 44454190 IC50 = 1995.26 nM T20251 C7H3CL 44454192 IC50 = 12589.25 nM T20251 CU0N1E 44454217 IC50 = 398.11 nM T20251 C9DBA3 44454218 IC50 = 12589.25 nM T20251 CK01QH 44454219 IC50 = 2511.89 nM T20251 CLO6X0 44454223 IC50 = 10000 nM T20251 CECR53 44454247 IC50 = 630.96 nM T20251 CD4ZU7 44454248 IC50 = 2511.89 nM T20251 CS2N1D 44454275 IC50 = 6309.57 nM T20251 CJ5XB1 44454278 IC50 = 63.1 nM T20251 C4GON0 44454309 IC50 = 6.31 nM T20251 C91PHS 44454318 IC50 = 1995.26 nM T20251 CT50UC 44454320 IC50 = 5011.87 nM T20251 C35WYK 44454339 IC50 = 2511.89 nM T20251 CZO96M 44454340 IC50 = 39810.72 nM T20251 C2CIO7 44454351 IC50 = 251.19 nM T20251 C9AH1O 44454352 IC50 = 794.33 nM T20251 CM8H2G 44454353 IC50 = 2511.89 nM T20251 C1EZP7 44454358 IC50 = 12589.25 nM T20251 CEB84V 44454371 IC50 = 50118.72 nM T20251 C5EV7Z 44454381 IC50 = 2511.89 nM T20251 CWC92Y 44454382 IC50 = 1584.89 nM T20251 CH0S2F 44454384 IC50 = 251.19 nM T20251 C32LHE 44454400 IC50 = 31622.78 nM T20251 CG18KC 44454401 IC50 = 251.19 nM T20251 CI0CJ9 44454402 IC50 = 50118.72 nM T20251 CP34QH 44454403 IC50 > 3981.07 nM T20251 CW4OX5 44454418 IC50 = 3162.28 nM T20251 CW1I4Z 44454420 IC50 = 12589.25 nM T20251 CXA7W2 44454458 IC50 = 398.11 nM T20251 CBGJ08 44454459 IC50 = 1258.93 nM T20251 C32WLZ 44454571 IC50 = 5700 nM T20251 C2Q0EH 44454597 IC50 = 6800 nM T20251 CL6KS1 44454834 IC50 > 3000 nM T20251 C6YQU9 44455589 Ki = 1590 nM T20251 C9PG3H 44455590 Ki = 7250 nM T20251 C1BR2G 44455619 Ki > 7500 nM T20251 CO1X6Z 44455620 Ki = 3751 nM T20251 C8F5CI 44455622 Ki = 3866 nM T20251 C4Z0WX 44455645 IC50 = 11000 nM T20251 C0EM9R 44455651 Ki = 1556 nM T20251 C3W1EZ 44455653 Ki = 2213 nM T20251 CI4K0E 44455654 Ki > 7500 nM T20251 CZV45C 44455655 Ki = 1757 nM T20251 C0L9YB 44455677 Ki > 7500 nM T20251 CV10IJ 44455678 Ki > 7500 nM T20251 CIW6A1 44455707 Ki = 5932 nM T20251 C3CXW8 44455739 Ki > 7500 nM T20251 CO4B1F 44455740 Ki = 4380 nM T20251 CBID06 44455782 IC50 = 12000 nM T20251 C02DNS 44456907 IC50 = 100000000 nM T20251 C3LQ5I 44456908 IC50 = 20417379.45 nM T20251 C05PZX 44456916 IC50 = 512861384 nM T20251 CG7E3Q 44456934 IC50 = 2951209.23 nM T20251 CB46NK 44456935 IC50 = 97723722.1 nM T20251 CVA46I 44456948 IC50 = 1412.54 nM T20251 COF1S4 44456951 IC50 = 85113803.82 nM T20251 CJ4NR1 44456970 IC50 = 645654229 nM T20251 CVB17U 44456974 IC50 = 66069344.8 nM T20251 CI71FO 44456993 IC50 = 446.68 nM T20251 C2MN1I 44456997 IC50 = 64565422.9 nM T20251 CT5H0R 44457009 IC50 = 100 nM T20251 C7VG4S 44457011 IC50 = 512861384 nM T20251 CNBT41 44457012 IC50 = 37153522.91 nM T20251 CX5IE3 44457029 IC50 = 758577575 nM T20251 CM0IE4 44457030 IC50 = 33113112.15 nM T20251 CTCQ07 44457046 IC50 = 81.28 nM T20251 C6HN4F 44457047 IC50 = 251188643.2 nM T20251 CRSI16 44457089 IC50 = 537031796.4 nM T20251 C2XZN7 44457090 IC50 = 45.71 nM T20251 CE6U0F 44457093 IC50 = 20.89 nM T20251 CW06YM 44457095 IC50 = 28183829.31 nM T20251 CPK1J7 44457105 IC50 = 2.512 nM T20251 CZEY35 44457108 IC50 = 43651583.22 nM T20251 CRPN60 44457141 IC50 = 158489319.3 nM T20251 CM65QS 44457156 IC50 = 6165950.02 nM T20251 CBSZ02 44458521 Ki = 43000 nM T20251 CIA6J1 44458523 Ki = 37000 nM T20251 C6LKZ7 44458534 Ki = 42000 nM T20251 CM65HC 44458548 Ki = 5300 nM T20251 CKM0F5 44458549 Ki = 6000 nM T20251 CC7I6Y 44458573 Ki = 73000 nM T20251 CF7I9V 44458586 Ki = 39000 nM T20251 CW7QX0 44458587 Ki = 16000 nM T20251 CJ7Y6A 44458592 Ki = 5500 nM T20251 C9QMB2 44458594 Ki > 90000 nM T20251 CPJW14 44458603 Ki > 90000 nM T20251 C0K2SV 44458617 Ki > 90000 nM T20251 CSIL15 44458629 Ki = 19000 nM T20251 C3EZ1V 44458770 Ki = 28000 nM T20251 CGT38B 44462719 Ki = 18000 nM T20251 CL9O8M 44462783 IC50 = 1970 nM T20251 C8WM0Z 44467183 IC50 = 44000 nM T20251 C5ETU8 44467185 IC50 = 19000 nM T20251 C7UDS1 44467360 IC50 = 1900 nM T20251 CQ0WM7 44469273 IC50 = 4200 nM T20251 C2KMI6 44469322 IC50 > 30000 nM T20251 C2QK4J 44472590 IC50 = 11200 nM T20251 CQ8C3F 44472591 IC50 = 2000 nM T20251 CC2TA5 44472592 IC50 > 30000 nM T20251 CWN95E 44472610 IC50 > 30000 nM T20251 C1H2ZT 44472612 IC50 > 30000 nM T20251 C9G5ID 44472613 IC50 > 30000 nM T20251 C5N4KE 44472633 IC50 > 30000 nM T20251 CJ39UE 44473168 Ki = 6800 nM T20251 C3CX0V 44475155 IC50 > 33000 nM T20251 C5RNK0 44476261 IC50 = 8600 nM T20251 CXY7T9 44476436 IC50 = 54200 nM T20251 C6V2YR 44476607 IC50 = 500 nM T20251 C6O0ZQ 44476624 IC50 = 34000 nM T20251 C6AK3W 44476911 IC50 > 30000 nM T20251 CLDQ43 44476913 IC50 > 30000 nM T20251 CG3R4T 44477000 IC50 = 14000 nM T20251 CDZP10 44479308 Ki = 950 nM T20251 CXJN29 44479309 Ki > 29000 nM T20251 C4Y5GO 44479310 Ki = 23000 nM T20251 CJDX78 44479549 IC50 > 10000 nM T20251 CJ25FS 44479563 Ki > 29000 nM T20251 C4CPX0 44479566 Ki = 15000 nM T20251 CI7EX6 44479809 Ki > 29000 nM T20251 C7C1HW 44481057 IC50 = 8100 nM T20251 C1FTA7 44481065 Ki > 29000 nM T20251 CVW53Z 44481067 Ki = 13000 nM T20251 C5COJ1 44481316 Ki = 4800 nM T20251 C8TIN9 44481318 Ki = 28000 nM T20251 CC2Q0J 44481321 Ki = 11000 nM T20251 C3NI0V 44481584 IC50 > 10000 nM T20251 C9U1KA 44481856 IC50 > 10000 nM T20251 CCA93X 44481857 IC50 > 10000 nM T20251 C13ZGK 44481860 Ki > 29000 nM T20251 CR3TH8 44481861 Ki = 17000 nM T20251 CW1ZR7 44481862 Ki = 7600 nM T20251 C8O9PY 44482139 Ki = 18000 nM T20251 CB0O7Y 44482409 Ki = 5000 nM T20251 C7XV2J 44512857 Ki = 28000 nM T20251 C5PI4H 44515310 Ki = 14 nM T20251 C1H8NX 44516817 IC50 > 30000 nM T20251 CFAZ41 44517710 IC50 = 16000 nM T20251 C68NXC 44517723 IC50 > 10000 nM T20251 C9OY3U 44517726 IC50 = 3162.28 nM T20251 C83JWO 44517778 IC50 = 3100 nM T20251 CS9H0L 44517795 IC50 > 100000 nM T20251 CSO35V 44520546 IC50 = 31622.78 nM T20251 C3Q5LP 44525560 IC50 = 3000 nM T20251 C9N1BU 44539192 IC50 > 15000 nM T20251 C01UWF 44540282 IC50 > 33000 nM T20251 CWP9Q3 44540283 IC50 = 17000 nM T20251 CKCG52 44540374 IC50 = 11000 nM T20251 C46HBA 44540470 IC50 = 23000 nM T20251 C2MF7Z 44540754 IC50 = 14000 nM T20251 C5O4TM 44540839 IC50 = 22000 nM T20251 CV92IJ 44541354 IC50 = 38.5 nM T20251 C6IK7J 44541892 IC50 = 33000 nM T20251 C16HIP 44542338 IC50 = 8700 nM T20251 C2B6OY 44542339 IC50 = 14100 nM T20251 CQ4W7V 44542340 IC50 = 14300 nM T20251 CD4LN9 44543781 IC50 = 21000 nM T20251 CS10AL 44543784 IC50 = 9300 nM T20251 C17LUC 44543889 IC50 = 14000 nM T20251 C9X2SL 44543890 IC50 = 26000 nM T20251 CE6HW8 44543891 IC50 > 33000 nM T20251 C27TZY 44543970 IC50 > 30000 nM T20251 CB83EJ 44544123 IC50 = 31000 nM T20251 CN64WQ 44544347 IC50 = 4600 nM T20251 CQ79RB 44544349 IC50 = 8600 nM T20251 CSV3F9 44544441 IC50 = 9200 nM T20251 C0RI5Z 44544444 IC50 = 7300 nM T20251 CK8T7U 44544546 IC50 = 8900 nM T20251 COJ7H6 44544644 IC50 = 5100 nM T20251 CYJB15 44544645 IC50 = 5500 nM T20251 C8RAF0 44544851 IC50 = 5500 nM T20251 CWKZ36 44544853 IC50 = 16000 nM T20251 C6AX2C 44544950 IC50 = 3300 nM T20251 CGB50M 44545053 IC50 = 9700 nM T20251 CU16DA 44545166 IC50 = 3600 nM T20251 CW78UO 44545168 IC50 = 4300 nM T20251 CNZ12F 44545169 IC50 = 5600 nM T20251 C5KZ2M 44545289 IC50 = 6600 nM T20251 C9JK4V 44545402 IC50 = 8200 nM T20251 C6L8QO 44545403 IC50 = 5600 nM T20251 CK1Z8P 44545482 IC50 > 30000 nM T20251 CX13MK 44547414 IC50 > 100000 nM T20251 CGLQ31 44552634 IC50 = 20000 nM T20251 CTX13C 44555196 IC50 = 16000 nM T20251 CUQ0J7 44555369 Ki > 13000 nM T20251 CJE2Q6 44555375 IC50 = 280 nM T20251 CT5N4E 44555481 IC50 = 11900 nM T20251 C4LJ6X 44557554 IC50 > 31600 nM T20251 C1EVH2 44560678 IC50 = 2143 nM T20251 CI58CZ 44560679 IC50 = 2500 nM T20251 CC4Z5M 44560681 IC50 = 10000 nM T20251 CWOM65 44560715 IC50 > 10000 nM T20251 C7YCO3 44560716 IC50 > 10000 nM T20251 C5X7PO 44560717 IC50 = 4800 nM T20251 COTH35 44560718 IC50 = 6100 nM T20251 C6J0ZC 44560719 IC50 = 7400 nM T20251 CL0A2D 44560720 IC50 = 3500 nM T20251 CR8K0X 44560724 IC50 = 9800 nM T20251 CE08JD 44560725 IC50 > 10000 nM T20251 CSX84T 44560726 IC50 = 9100 nM T20251 C1O0IG 44560727 IC50 = 6000 nM T20251 CB7X4S 44560728 IC50 = 8300 nM T20251 C94LIO 44560729 IC50 > 10000 nM T20251 C3UQ8C 44560730 IC50 > 10000 nM T20251 C8OD4F 44560731 IC50 = 4700 nM T20251 CLB20U 44560732 IC50 > 10000 nM T20251 CC01KM 44561020 IC50 = 13000 nM T20251 C4SVU2 44561370 IC50 = 740 nM T20251 CRJM24 44561454 IC50 = 7800 nM T20251 CXJK43 44561493 IC50 = 13000 nM T20251 CY14MD 44561518 IC50 = 86 nM T20251 CR8OX1 44562611 IC50 = 1780 nM T20251 CL64BM 44562612 IC50 = 2110 nM T20251 CVB0Q6 44562613 IC50 = 3040 nM T20251 C02CWF 44562614 IC50 = 2110 nM T20251 C7CSF8 44562615 IC50 = 873 nM T20251 CNJM41 44562616 IC50 = 1230 nM T20251 C3VP6N 44562943 IC50 = 1740 nM T20251 C7DS0M 44562944 IC50 = 10400 nM T20251 C4XL2E 44562989 IC50 = 3880 nM T20251 C5J6HU 44563054 IC50 = 3010 nM T20251 CZW0B1 44563061 IC50 = 4700 nM T20251 CT9S4L 44563063 IC50 = 460 nM T20251 C2HJ9Z 44563066 IC50 = 7000 nM T20251 C83CZN 44563067 IC50 > 32000 nM T20251 C97AJO 44563111 IC50 = 20000 nM T20251 CL3MW0 44563112 IC50 = 11000 nM T20251 C6B2FI 44563127 IC50 = 4800 nM T20251 CL0DS9 44563128 IC50 = 5440 nM T20251 CDTB89 44563137 IC50 = 350 nM T20251 C51TLU 44563144 IC50 = 10000 nM T20251 CNR1B2 44563145 IC50 = 3000 nM T20251 C0D1LO 44563146 IC50 = 20000 nM T20251 C0J2GS 44563163 IC50 = 3210 nM T20251 C67TOD 44563164 IC50 = 3030 nM T20251 CL5HW8 44563165 IC50 = 2690 nM T20251 CJV9S8 44563177 IC50 = 6000 nM T20251 CV90NH 44563178 IC50 > 32000 nM T20251 CDX3R8 44563203 IC50 = 785 nM T20251 C5QX2S 44563204 IC50 = 5110 nM T20251 CF4ZK8 44563205 IC50 = 1640 nM T20251 C3ZUH6 44563206 IC50 = 1150 nM T20251 CJ9O6U 44563238 IC50 = 645 nM T20251 CB8P3I 44563239 IC50 = 3690 nM T20251 CB9NG8 44563240 IC50 = 2470 nM T20251 CN5U4V 44563241 IC50 = 5230 nM T20251 CLJ7C2 44563242 IC50 = 3120 nM T20251 C2OX9D 44563243 IC50 = 4790 nM T20251 C1VQ5X 44563244 IC50 = 1060 nM T20251 CU9J5W 44564565 IC50 > 100000 nM T20251 C3MNR0 44565080 IC50 > 10000 nM T20251 CF6JG1 44565081 IC50 > 10000 nM T20251 CA0FC1 44565082 IC50 = 2300 nM T20251 C6DI0T 44565083 IC50 = 2100 nM T20251 CV1IL5 44565796 IC50 = 70000 nM T20251 C9SL5D 44565872 IC50 > 10000 nM T20251 COA7X5 44565892 IC50 = 54000 nM T20251 C3YE7P 44567441 IC50 = 11 nM T20251 C46KUB 44568231 IC50 = 1200 nM T20251 COTQ47 44568792 IC50 = 3034 nM T20251 CWLT20 44570180 IC50 > 63000 nM T20251 C1W9AF 44570584 IC50 = 15700 nM T20251 CXHT91 44571305 IC50 = 6000 nM T20251 CR32XZ 44571307 IC50 = 17000 nM T20251 CIV48S 44572053 IC50 = 2018 nM T20251 CZM8O6 44573159 Ki = 3410 nM T20251 CVSJ62 44573160 Ki = 3690 nM T20251 CF0A2J 44573161 Ki = 2090 nM T20251 C13LFI 44573162 Ki = 3430 nM T20251 C7HZJ6 44573224 Ki = 5240 nM T20251 CO4NI2 44573249 Ki = 17 nM T20251 C9OF8P 44573250 Ki = 169 nM T20251 CPJ27Z 44573251 Ki = 35 nM T20251 CIK5T2 44573291 Ki = 201 nM T20251 CM89KA 44573292 Ki = 82 nM T20251 CI6F0Y 44573293 Ki = 343 nM T20251 CL6C7B 44573294 Ki = 548 nM T20251 CBM82T 44573332 Ki > 10000 nM T20251 CMSV07 44573403 Ki = 1840 nM T20251 CLX14F 44573404 Ki > 10000 nM T20251 C0PD8L 44573405 Ki = 9690 nM T20251 CA03TK 44573444 Ki > 10000 nM T20251 CZ26TO 44573445 Ki = 865 nM T20251 CQ9WA5 44573446 Ki = 518 nM T20251 CKJ2O8 44573447 Ki = 746 nM T20251 CNUJ50 44574003 IC50 > 10000 nM T20251 C1T4QN 44574053 IC50 = 2000 nM T20251 C5LJ0D 44577963 IC50 = 1380 nM T20251 CFJB16 44578266 Ki > 2700 nM T20251 CML90U 44578389 IC50 = 710 nM T20251 CD1U2S 44578570 IC50 = 5500 nM T20251 C1MC0I 44578615 IC50 = 18000 nM T20251 CFAW91 44578616 IC50 = 8400 nM T20251 CYPJ70 44578617 IC50 > 24000 nM T20251 CR0F7I 44578649 IC50 > 32000 nM T20251 C9E6QP 44579079 IC50 = 5770 nM T20251 C7CKG9 44579080 IC50 = 1455 nM T20251 CH5B0N 44579120 IC50 = 420 nM T20251 CN42GY 44579121 IC50 = 710 nM T20251 CDUJ10 44579122 IC50 = 360 nM T20251 CQJ0L6 44579123 IC50 = 540 nM T20251 CO13BP 44579170 IC50 = 890 nM T20251 CP0X4D 44579171 IC50 = 2340 nM T20251 CS60PG 44579172 IC50 = 5040 nM T20251 CY2E6M 44579173 IC50 > 30000 nM T20251 C4RNV0 44580338 Ki = 26 nM T20251 CE87QS 44580381 Ki = 94 nM T20251 C9B2LH 44580383 Ki = 49 nM T20251 C3L5ER 44583033 IC50 = 11800 nM T20251 CTO9G3 44583367 IC50 > 30000 nM T20251 CL62PK 44588589 IC50 = 198 nM T20251 CMI7N1 44588590 IC50 = 680 nM T20251 CP9QH1 44588591 IC50 = 71500 nM T20251 CLZ05M 44588592 IC50 = 740 nM T20251 C09TKD 44589077 IC50 = 31800 nM T20251 CKU85Z 44589520 Ki = 14560 nM T20251 C9RA0C 44589548 EC50 > 30000 nM T20251 CT7F0N 44589856 Ki = 590 nM T20251 C3C6WU 44589911 Ki = 19250 nM T20251 CVA4I9 44589912 Ki > 10000 nM T20251 CVQ83W 44589913 Ki = 9800 nM T20251 CNBO74 44589970 EC50 = 3300 nM T20251 C0GQ2C 44589971 Ki = 760 nM T20251 C9OL3W 44590015 Ki = 1900 nM T20251 C5AWD8 44590016 Ki = 170 nM T20251 C0MLS4 44590017 Ki = 3200 nM T20251 CGP0W8 44590018 Ki = 97 nM T20251 C4C5AQ 44590111 Ki = 6300 nM T20251 CVZ23T 44590151 Ki > 10000 nM T20251 CDC86A 44590152 Ki = 9420 nM T20251 CJ0U5K 44590153 Ki = 8620 nM T20251 CB67HK 44590208 Ki = 10980 nM T20251 CRG54L 44590209 Ki = 8699 nM T20251 C1G2VQ 44590210 Ki = 9070 nM T20251 CJK1Q3 44590211 Ki = 7540 nM T20251 CU71HW 44590230 IC50 = 849 nM T20251 CE5U9X 44590439 IC50 = 3410 nM T20251 CS8ZR6 44590583 IC50 = 248 nM T20251 CRN4U5 44590696 IC50 = 86000 nM T20251 CIH56J 44590864 IC50 = 4.7 nM T20251 CZ5HT9 44590865 IC50 = 117 nM T20251 CAC12Y 44590943 IC50 = 3100 nM T20251 C2EB4O 44590944 IC50 < 5280 nM T20251 CHQM54 44590946 IC50 = 1650 nM T20251 C1OCI9 44591315 IC50 = 237 nM T20251 C7GL4H 44591704 Ki = 1020 nM T20251 C91FTW 44591848 IC50 = 85000 nM T20251 CY78PR 44591849 IC50 = 55000 nM T20251 CE2LW5 44591850 IC50 = 59000 nM T20251 CI6R1Z 44592120 Ki = 4500 nM T20251 C1QO8J 44592121 Ki = 10300 nM T20251 CVT6R5 44592123 Ki = 716 nM T20251 CV8E7O 44592155 Ki = 412 nM T20251 CMS5I2 44592158 Ki > 5000 nM T20251 C4EH6O 44592207 Ki = 100 nM T20251 CZ5I1N 44592208 Ki = 3162.28 nM T20251 CKM8T7 44592209 Ki = 7943.28 nM T20251 CJO9K5 44592245 Ki = 10100 nM T20251 CDJ32U 44592249 Ki = 5011.87 nM T20251 CS2FL4 44592250 Ki = 1584.89 nM T20251 CL17WU 44592251 Ki = 1584.89 nM T20251 CJCL64 44592252 Ki = 398.11 nM T20251 CO6ES5 44592257 IC50 = 7300 nM T20251 CM0I3E 44592294 Ki = 10000 nM T20251 CQ04EG 44592295 Ki = 12589.25 nM T20251 C65XQL 44592296 Ki = 3981.07 nM T20251 CEB2S1 44592297 Ki = 3162.28 nM T20251 CP51QS 44592332 Ki = 5011.87 nM T20251 CD2Z4J 44592333 Ki = 6309.57 nM T20251 C7NCT2 44592334 Ki = 6309.57 nM T20251 CHY20X 44592335 Ki = 3162.28 nM T20251 C5H7XK 44592371 Ki = 630.96 nM T20251 CI7G1T 44592534 IC50 = 7800.01 nM T20251 C69VSL 44592535 IC50 = 6000 nM T20251 COE58F 44592580 IC50 = 190 nM T20251 CP1U5K 44592598 IC50 = 1100 nM T20251 CCQ73Z 44592962 IC50 = 5800 nM T20251 C6HA0L 44592987 IC50 = 50000 nM T20251 CDP7R8 44592988 IC50 = 50000 nM T20251 CE62VG 44592989 IC50 = 20999.99 nM T20251 C21FGX 44592990 IC50 = 11000.01 nM T20251 CUX2C0 44593418 IC50 = 88 nM T20251 CDC59A 44593419 IC50 = 135 nM T20251 CSD5Z3 44593420 IC50 = 1930 nM T20251 CQ12YR 44593444 IC50 = 2120 nM T20251 C2U5KV 44593866 IC50 > 1000 nM T20251 CKTZ17 44594174 IC50 = 52000 nM T20251 C3CJW9 44595244 Ki = 637 nM T20251 C96MTQ 44595526 Ki = 5214 nM T20251 CF4YN8 44598057 IC50 = 1905.46 nM T20251 C9MT0V 44598058 IC50 = 1905.46 nM T20251 C71QNY 44598059 IC50 = 229.09 nM T20251 C9TH0G 44598060 IC50 = 11220.18 nM T20251 CZWY54 44598061 IC50 = 19498.45 nM T20251 CP27OH 44598062 IC50 = 38018.94 nM T20251 CS76XZ 44598121 IC50 = 16982.44 nM T20251 C0L4FZ 44598124 IC50 = 30902.95 nM T20251 CGQT32 44598769 IC50 = 19054.61 nM T20251 CG2SD8 44598819 IC50 = 2344.23 nM T20251 C27GZB 44598820 IC50 = 5128.61 nM T20251 CV9G1H 44598821 IC50 = 70.79 nM T20251 CM2UG7 44598902 IC50 = 6000 nM T20251 C84NFS 44599828 IC50 = 2400 nM T20251 CVJG25 44600846 IC50 = 4600 nM T20251 C89VRG 44605616 IC50 > 50118.72 nM T20251 CZD25I 44605617 IC50 > 50118.72 nM T20251 CEQN62 44609163 IC50 > 30000 nM T20251 C7G4FT 44609164 IC50 > 30000 nM T20251 CH9FO5 44609165 IC50 > 30000 nM T20251 CLPY85 44609168 IC50 > 30000 nM T20251 CU0QT2 44609322 IC50 = 23000 nM T20251 CQ06VN 44609327 IC50 > 30000 nM T20251 CE9GN6 44609485 IC50 > 30000 nM T20251 C9GWF1 44609645 IC50 = 7000 nM T20251 CI10GR 44610722 Ki = 1600 nM T20251 CW84TH 44610723 Ki = 3200 nM T20251 CPIB93 44610724 Ki = 11000 nM T20251 CDX2H1 44621189 IC50 = 15800 nM T20251 CO3I5F 44622849 Ki > 22000 nM T20251 C8B0HO 44622872 IC50 = 396 nM T20251 CZHP95 44626357 IC50 = 3700 nM T20251 C9N4MQ 44626527 IC50 = 1995.26 nM T20251 CSJ9F1 44626530 IC50 = 630.96 nM T20251 CCLQ67 44626632 IC50 = 794.33 nM T20251 CA93OY 44626637 IC50 = 251.19 nM T20251 CPML65 44626639 IC50 = 125.89 nM T20251 CDA90T 44626641 IC50 = 630.96 nM T20251 C2TBL0 44626734 IC50 = 630.96 nM T20251 C7LUV5 44626738 IC50 = 630.96 nM T20251 CRCL97 44626740 IC50 = 199.53 nM T20251 CZ25SY 44626744 IC50 = 630.96 nM T20251 C5DM7T 44626835 IC50 = 251.19 nM T20251 C85ZIF 44626928 IC50 = 158.49 nM T20251 C4BYG5 44626929 IC50 = 1000 nM T20251 CK5BG2 44626935 IC50 = 630.96 nM T20251 CWL84Q 44627022 IC50 = 1584.89 nM T20251 CGXJ71 44627023 IC50 = 630.96 nM T20251 CBP18J 44627024 IC50 = 398.11 nM T20251 C30KEM 44627025 IC50 = 398.11 nM T20251 CV1DO3 44627033 IC50 = 1258.93 nM T20251 CAH6O1 44627120 IC50 = 3981.07 nM T20251 CUE56O 44627123 IC50 = 110 nM T20251 CDY32E 44627127 IC50 = 1258.93 nM T20251 CJ4ZQ0 44627129 IC50 = 1995.26 nM T20251 CN1O6P 44627131 IC50 = 1000 nM T20251 CQE59L 44627133 IC50 = 3162.28 nM T20251 C4QV9Y 44627238 IC50 = 6309.57 nM T20251 C1D5FJ 44627240 IC50 = 199.53 nM T20251 CNK4P0 44627242 IC50 = 501.19 nM T20251 CY3LE2 44627245 IC50 = 398.11 nM T20251 C5LN9E 44627351 IC50 = 501.19 nM T20251 CLUN07 44627353 IC50 = 1258.93 nM T20251 CZ1FY5 44627355 IC50 = 3162.28 nM T20251 C3ZWA4 44627357 IC50 = 630.96 nM T20251 CY1TE0 44627358 IC50 = 1995.26 nM T20251 CG97OK 44627359 IC50 = 1000 nM T20251 C65RAG 44627466 IC50 = 1000 nM T20251 C06TJC 44627468 IC50 = 398.11 nM T20251 CBV8I6 44627470 IC50 = 1258.93 nM T20251 C7NIU3 44628133 IC50 = 50 nM T20251 CE6M8G 44628198 IC50 = 9960 nM T20251 CERD02 44628200 IC50 = 20 nM T20251 CIM8C4 44628201 IC50 = 10 nM T20251 C1XQ8G 44629350 IC50 = 1220 nM T20251 CMO1Z6 44631854 IC50 > 30000 nM T20251 CIX15W 44631974 IC50 > 90000 nM T20251 C37AQP 44815590 IC50 = 8500 nM T20251 CU8P7K 44815806 Ki = 28540 nM T20251 C4C9LB 44815976 Ki = 2500 nM T20251 C0LRQ2 45101475 IC50 = 19000 nM T20251 CSEP-69 45102708 IC50 > 15848.93 nM T20251 C32YHG 45102733 Ki = 200 nM T20251 C45PUQ 45102745 Ki = 4200 nM T20251 C4XAC1 45103619 IC50 > 30000 nM T20251 C4G7PQ 45104756 IC50 = 5740 nM T20251 CVCQ85 45104767 IC50 = 95000 nM T20251 C0DLU3 45109862 IC50 = 100 nM T20251 C40BIM 45139151 IC50 = 17700 nM T20251 C4KRT0 45254002 IC50 = 29300 nM T20251 CJ0Y1O 45254127 Ki > 10000 nM T20251 C8FQ9P 45254130 Ki > 10000 nM T20251 CQB45G 45254505 Ki > 10000 nM T20251 C1R3PL 45254506 Ki > 10000 nM T20251 C2JD1Y 45254508 Ki > 10000 nM T20251 C2YE7A 45254510 Ki > 10000 nM T20251 C2M9RC 45254900 Ki = 3280 nM T20251 CUL8G3 45255106 Ki > 15000 nM T20251 C43HDC 45256109 Ki = 660 nM T20251 C2Q3MJ 45256294 Ki = 1840 nM T20251 C5RQ2B 45256296 Ki = 410 nM T20251 C0Q2WV 45256478 Ki = 4980 nM T20251 C8H4SQ 45256479 Ki > 15000 nM T20251 CV32EW 45256653 Ki = 10700 nM T20251 C5LYK1 45256654 Ki = 1420 nM T20251 CE9IU1 45256823 Ki = 150 nM T20251 CI70YH 45256826 Ki = 1160 nM T20251 CT41IW 45256827 Ki > 15000 nM T20251 C1K0ZH 45259193 IC50 = 2511.89 nM T20251 C0C4FV 45265850 IC50 > 14000 nM T20251 CAHW68 45267251 IC50 = 5011.87 nM T20251 CW1S6B 45267254 IC50 = 3162.28 nM T20251 CD47IO 45267261 IC50 = 794.33 nM T20251 CJPS81 45267262 IC50 = 1995.26 nM T20251 C4HOR6 45267270 IC50 = 1995.26 nM T20251 CUT2B4 45267348 IC50 > 30000 nM T20251 CF4PM0 45267382 IC50 = 900 nM T20251 C1N5ZL 45267385 IC50 = 800 nM T20251 C4AZD3 45267386 IC50 = 3500 nM T20251 C8LPF5 45267399 IC50 = 2340 nM T20251 C8PR5X 45267430 IC50 > 31600 nM T20251 C3T5PI 45267459 IC50 = 2900 nM T20251 CPD18Y 45267471 IC50 = 12589.25 nM T20251 CL0WP4 45267480 IC50 = 63.1 nM T20251 C2H4ZX 45267491 IC50 = 794.33 nM T20251 C0KTX2 45267492 IC50 = 794.33 nM T20251 C2R9HN 45267503 IC50 = 2511.89 nM T20251 CEY87M 45267504 IC50 = 1584.89 nM T20251 CFY4R2 45267593 IC50 > 10000 nM T20251 CP7XE6 45267597 IC50 > 10000 nM T20251 CK58HY 45267611 IC50 = 9210 nM T20251 CM23AU 45267709 IC50 = 19600 nM T20251 CGB32I 45267714 IC50 = 3080 nM T20251 CO3Y0N 45267724 IC50 > 31600 nM T20251 CI7KZ2 45267735 IC50 = 5340 nM T20251 CC5OP0 45267739 IC50 = 12700 nM T20251 CXJ8H3 45267746 IC50 = 25800 nM T20251 CUEY48 45267808 IC50 = 14600 nM T20251 CF2R3T 45268112 IC50 = 1584.89 nM T20251 C3S5ZP 45268113 IC50 = 630.96 nM T20251 C0UG9Z 45268119 IC50 = 19952.62 nM T20251 C37TAV 45268120 IC50 = 1000 nM T20251 CP1TV2 45268127 IC50 = 31622.78 nM T20251 C79VFY 45268141 IC50 = 3981.07 nM T20251 C64NZQ 45268142 IC50 = 25118.86 nM T20251 CENZ75 45268148 IC50 = 6309.57 nM T20251 CJH3A2 45268206 IC50 > 30000 nM T20251 CTB32R 45268225 IC50 = 400 nM T20251 CP85WO 45268247 IC50 = 31000 nM T20251 C0XAR6 45268283 IC50 = 12 nM T20251 C7V1WF 45268290 IC50 = 4.4 nM T20251 C9RCS2 45268299 IC50 = 1000 nM T20251 CLF90U 45268300 IC50 = 1700 nM T20251 C2T0ZC 45268315 IC50 = 1300 nM T20251 CM1SA7 45268333 IC50 = 1000 nM T20251 CH53XO 45268345 IC50 = 7.943 nM T20251 CHB5U0 45268346 IC50 = 251.19 nM T20251 COCN89 45268373 IC50 = 6309.57 nM T20251 C4MU3C 45268438 IC50 = 3162.28 nM T20251 C4DZO1 45268459 IC50 > 10000 nM T20251 CRP90V 45268466 IC50 > 16300 nM T20251 CQ7J4A 45268477 IC50 > 10000 nM T20251 CSJ4L2 45268478 IC50 > 20000 nM T20251 C9IJK8 45268483 IC50 = 7400 nM T20251 C7UG6Q 45268498 IC50 = 15000 nM T20251 C7VZR5 45268637 IC50 = 20900 nM T20251 CV1IR5 45268644 IC50 > 31600 nM T20251 C9B5EH 45268653 Ki = 116 nM T20251 C18EGU 45268687 IC50 = 530 nM T20251 CUQ23Z 45268922 IC50 > 10000 nM T20251 CEK21M 45268987 IC50 = 10000 nM T20251 CHB76Z 45268990 IC50 = 3981.07 nM T20251 CR3YU9 45268999 IC50 = 3981.07 nM T20251 CW57CP 45269000 IC50 = 7943.28 nM T20251 CYQ1I7 45269020 IC50 = 199.53 nM T20251 C4WR0V 45269087 IC50 > 30000 nM T20251 CRPS25 45269096 IC50 = 27000 nM T20251 C7BNY6 45269104 IC50 = 6000 nM T20251 CC8P5K 45269117 IC50 = 480 nM T20251 C6ETI8 45269118 IC50 = 910 nM T20251 CX53RU 45269119 IC50 = 7000 nM T20251 CRN8Y1 45269121 IC50 = 1600 nM T20251 CVH8S4 45269235 IC50 = 3162.28 nM T20251 CED18G 45269300 IC50 > 10000 nM T20251 CZC09M 45269305 IC50 > 10000 nM T20251 CFJ17A 45269306 IC50 > 10000 nM T20251 CCQ8W4 45269310 IC50 = 6700 nM T20251 CNA70T 45269316 IC50 > 10000 nM T20251 C1SB8A 45269317 IC50 > 10000 nM T20251 C5OED7 45269318 IC50 > 20000 nM T20251 CF2P9H 45269325 IC50 > 20000 nM T20251 CQ03ZU 45269337 IC50 > 20000 nM T20251 CXE36D 45269351 IC50 > 7460 nM T20251 C78UOX 45269357 IC50 = 9900 nM T20251 C4WT5J 45269358 IC50 = 15000 nM T20251 C97ZET 45269449 IC50 = 780 nM T20251 CU02ZQ 45269860 IC50 = 1995.26 nM T20251 CS1Q2X 45269947 IC50 > 30000 nM T20251 C1BE5U 45269948 IC50 > 30000 nM T20251 CG1H9N 45269950 IC50 = 8200 nM T20251 CA3MZ6 45269996 IC50 = 14000 nM T20251 C5DIS2 45270014 IC50 = 1000 nM T20251 C8C2AK 45270025 IC50 = 25 nM T20251 C2L8JN 45270044 IC50 = 7000 nM T20251 CDM73H 45270136 IC50 = 2100 nM T20251 C2Q4SM 45270142 IC50 > 10000 nM T20251 CX31KD 45270149 IC50 = 1440 nM T20251 CLPB92 45270153 IC50 = 9000 nM T20251 CGXC75 45270156 IC50 > 10000 nM T20251 C3GA6N 45270158 IC50 > 18200 nM T20251 C3KI7Q 45270163 IC50 > 20000 nM T20251 C0QR1E 45270171 IC50 > 17600 nM T20251 C6YI5N 45270172 IC50 > 18500 nM T20251 CZ9DA3 45270173 IC50 = 2350 nM T20251 CA38NB 45270184 IC50 = 31000 nM T20251 CPG7D6 45270273 IC50 > 31600 nM T20251 C0J6BO 45270297 IC50 > 31600 nM T20251 C23PMF 45270302 IC50 > 31600 nM T20251 C9WNG1 45270303 IC50 = 7330 nM T20251 C4SXQ3 45270319 IC50 = 6900 nM T20251 C8GQ7J 45270330 Ki = 1461 nM T20251 C48BMQ 45270339 Ki > 7500 nM T20251 CS67XW 45270376 IC50 = 460 nM T20251 COFD89 45270589 IC50 = 6610 nM T20251 CEX26T 45270595 IC50 = 950 nM T20251 CF43XE 45270678 IC50 = 31622.78 nM T20251 CK01NU 45270702 IC50 = 12589.25 nM T20251 C1NT2M 45270771 IC50 > 30000 nM T20251 CA05IG 45270778 IC50 = 9000 nM T20251 CZ7MK9 45270788 IC50 = 7000 nM T20251 C0R5NB 45270796 IC50 = 4300 nM T20251 C3A0NB 45270802 IC50 = 630 nM T20251 C35TNH 45270803 IC50 = 1090 nM T20251 C3GLV8 45270841 IC50 = 2170 nM T20251 CD5OS6 45270850 IC50 > 31600 nM T20251 CUV67Q 45270855 IC50 = 11 nM T20251 C5UP2J 45270862 IC50 = 470 nM T20251 CEM4Z0 45270863 IC50 = 6300 nM T20251 C9GK5C 45270870 IC50 = 4800 nM T20251 CO0P8H 45270903 IC50 = 398.11 nM T20251 C7OM4D 45270916 IC50 = 50118.72 nM T20251 CZ9OC8 45270973 IC50 = 530 nM T20251 CB94YA 45270992 IC50 = 4700 nM T20251 C13QSU 45270993 IC50 > 16800 nM T20251 CU9HV3 45271001 IC50 = 2210 nM T20251 CBW87K 45271004 IC50 = 1300 nM T20251 C71AON 45271011 IC50 > 19000 nM T20251 C2G5XK 45271015 IC50 = 19000 nM T20251 CO05CL 45271041 IC50 = 3200 nM T20251 C42GYR 45271095 IC50 = 1810 nM T20251 C1F5RT 45271103 IC50 = 3000 nM T20251 CCN0F4 45271111 IC50 = 11700 nM T20251 CS9M8B 45271114 IC50 = 4120 nM T20251 CY70FL 45271134 IC50 = 1300 nM T20251 C18WQE 45271166 Ki > 5000 nM T20251 CMQ25P 45271491 IC50 = 1000 nM T20251 CEQ19M 45271499 IC50 = 2511.89 nM T20251 CESN63 45271510 IC50 = 1584.89 nM T20251 CMDC23 45271511 IC50 = 15848.93 nM T20251 C8TXI5 45271516 IC50 = 6309.57 nM T20251 C5P3FX 45271520 IC50 = 1584.89 nM T20251 CF9I3G 45271548 IC50 = 794.33 nM T20251 C9TM2P 45271593 IC50 > 30000 nM T20251 C06YAD 45271599 IC50 > 30000 nM T20251 CG0I8P 45271610 IC50 > 30000 nM T20251 C6FBH0 45271618 IC50 = 2600 nM T20251 C08OEP 45271626 IC50 = 830 nM T20251 C13PCQ 45271633 IC50 = 1600 nM T20251 C3OA8C 45271642 IC50 = 1550 nM T20251 CP7CX1 45271647 IC50 = 28000 nM T20251 CH1PS3 45271663 IC50 > 31600 nM T20251 CM4ZX1 45271673 IC50 = 1700 nM T20251 CN4W1B 45271701 IC50 = 440 nM T20251 CW0JQ7 45271712 IC50 = 2500 nM T20251 CAO92B 45271713 IC50 = 14000 nM T20251 C6R3LQ 45271737 IC50 = 1258.93 nM T20251 CM5Q8S 45271738 IC50 = 63.1 nM T20251 C42EJD 45271753 IC50 = 2511.89 nM T20251 CT3DP1 45271760 IC50 = 1584.89 nM T20251 CE8Z1K 45271821 IC50 = 520 nM T20251 C1L4DN 45271828 IC50 > 10000 nM T20251 CLD3T9 45271838 IC50 > 10000 nM T20251 C1S6TI 45271840 IC50 > 20000 nM T20251 C3QAP5 45271853 IC50 > 20000 nM T20251 CP7K0V 45271861 IC50 > 10000 nM T20251 CFG5Z3 45271864 IC50 > 20000 nM T20251 C36SRE 45271994 IC50 = 3870 nM T20251 C73LNM 45272006 IC50 = 3330 nM T20251 CMYT82 45272014 IC50 = 4890 nM T20251 C60DPZ 45272024 IC50 > 31600 nM T20251 C2MKZ1 45272040 IC50 > 31600 nM T20251 CU9C4I 45272046 Ki = 40 nM T20251 CAY8I7 45272070 Ki = 3536 nM T20251 C5U7LD 45272411 IC50 = 10000 nM T20251 CM9W5B 45272412 IC50 = 25118.86 nM T20251 CG9CO5 45272414 IC50 = 6309.57 nM T20251 C4W9NG 45272415 IC50 = 398.11 nM T20251 C12WFN 45272425 IC50 = 1258.93 nM T20251 CK67XC 45272426 IC50 = 3162.28 nM T20251 CQ2ZS6 45272434 IC50 = 12589.25 nM T20251 CGKZ21 45272435 IC50 = 19952.62 nM T20251 CH0MA8 45272437 IC50 = 63095.73 nM T20251 CW2MD0 45272438 IC50 = 3981.07 nM T20251 C71VIG 45272510 IC50 = 2000 nM T20251 C05EDY 45272511 IC50 = 27000 nM T20251 C5R7OL 45272520 IC50 = 540 nM T20251 C6FCW0 45272539 IC50 = 10000 nM T20251 CGV7P0 45272576 IC50 = 5 nM T20251 CR1F7A 45272583 IC50 = 1300 nM T20251 C1TLM4 45272592 IC50 = 3800 nM T20251 CE1P8L 45272616 IC50 = 1258.93 nM T20251 CEO57P 45272634 IC50 = 3162.28 nM T20251 CI7C1L 45272635 IC50 = 6309.57 nM T20251 C5DE4U 45272692 IC50 = 9600 nM T20251 CN3G7M 45272695 Ki = 130000 nM T20251 CPM1U3 45272720 IC50 > 20000 nM T20251 CJ52PS 45272816 IC50 = 2030 nM T20251 CT5KW9 45272826 IC50 = 6500 nM T20251 CD6FR7 45272837 IC50 = 2160 nM T20251 C3GUS5 45272853 IC50 > 31600 nM T20251 C62IGT 45272875 Ki = 57 nM T20251 C3GUK4 45272876 Ki = 73 nM T20251 CBE0M8 45272877 Ki = 158 nM T20251 CR04WH 45272878 Ki = 102 nM T20251 CZ7N8Q 45272889 Ki = 426 nM T20251 CK2B5U 45272890 Ki = 776 nM T20251 C8TC4R 45272894 Ki = 137 nM T20251 CA0SD1 45272895 IC50 = 809 nM T20251 CH17KU 45272913 IC50 = 65600 nM T20251 CPUR70 45272936 IC50 = 2200 nM T20251 CQ98IX 45272939 IC50 = 3800 nM T20251 CX1QY9 45273266 IC50 = 3162.28 nM T20251 C62LGY 45273272 IC50 = 1995.26 nM T20251 CZ2OL1 45273273 IC50 = 7943.28 nM T20251 CBM9R2 45273292 IC50 = 1258.93 nM T20251 CS04AC 45273293 IC50 = 15848.93 nM T20251 CS95IU 45273334 IC50 = 5011.87 nM T20251 CD62AH 45273373 IC50 > 30000 nM T20251 CMN39U 45273380 IC50 = 10000 nM T20251 C9JQT2 45273392 IC50 = 1020 nM T20251 CPTE06 45273401 IC50 = 11700 nM T20251 CG4YS2 45273406 IC50 = 4200 nM T20251 C0GK4R 45273485 IC50 = 6200 nM T20251 CFY94G 45273510 IC50 = 5011.87 nM T20251 CRSF80 45273522 IC50 = 1584.89 nM T20251 C3DB8P 45273523 IC50 = 199.53 nM T20251 CM10UD 45273529 IC50 = 79.43 nM T20251 CRD9C8 45273530 IC50 = 630.96 nM T20251 CNQJ09 45273545 IC50 = 1995.26 nM T20251 C7XC3T 45273551 IC50 = 3981.07 nM T20251 C1JLQ3 45273630 IC50 > 10000 nM T20251 C27VWT 45273649 IC50 = 900 nM T20251 C7HQ9B 45273656 IC50 > 10000 nM T20251 CT3V0B 45273663 IC50 > 13500 nM T20251 C58HQB 45273679 IC50 = 34000 nM T20251 CLFN69 45273777 IC50 = 4700 nM T20251 CP7OZ1 45273778 IC50 = 14700 nM T20251 COD72W 45273783 IC50 = 7930 nM T20251 CCJR41 45273790 IC50 = 3960 nM T20251 C3TZ8X 45273801 IC50 = 4040 nM T20251 CX9T5I 45273802 IC50 = 2840 nM T20251 C5E2XR 45273828 Ki = 157 nM T20251 CN4IE3 45275362 IC50 > 100000 nM T20251 C2GKC7 45278576 IC50 > 80000 nM T20251 C2J0GO 45278647 IC50 = 6800 nM T20251 CZ71RN 45278805 IC50 = 140 nM T20251 CZN6M7 45278882 IC50 = 540 nM T20251 C3NW0C 45279216 IC50 = 500 nM T20251 C7DXG1 45279490 IC50 = 5500 nM T20251 CR0N4Z 45279585 IC50 = 3000 nM T20251 C7XI9W 45279680 IC50 > 10000 nM T20251 C84XIH 45279772 IC50 = 3300 nM T20251 CJO30G 45279869 IC50 = 2000 nM T20251 CLX86A 45380509 IC50 = 11000 nM T20251 CL41HJ 45380693 IC50 = 3200 nM T20251 C9NCV4 45380694 IC50 = 3700 nM T20251 C6SZ8A 45380791 IC50 = 4800 nM T20251 CEM0V9 45380893 IC50 = 10000 nM T20251 CU7Z8X 45381216 IC50 > 33000 nM T20251 CWA35Y 45381330 IC50 = 16000 nM T20251 C5I3OG 45381546 IC50 = 5900 nM T20251 C9UF1Z 45381640 IC50 > 33000 nM T20251 CP3HD2 45381723 IC50 > 33000 nM T20251 C4AM7K 45381799 IC50 = 9100 nM T20251 CG1QY5 45381801 IC50 = 4600 nM T20251 CO4BT1 45381802 IC50 = 2700 nM T20251 CT21WU 45381890 IC50 = 12000 nM T20251 CWJM09 45381983 IC50 > 33000 nM T20251 C91UWI 45482679 IC50 = 204.08 nM T20251 CP1YN5 45482680 IC50 = 1363.64 nM T20251 CV56HF 45482684 IC50 = 6949.15 nM T20251 C2C1XZ 45482685 IC50 = 204.08 nM T20251 CA45ZR 45482686 IC50 = 2658.23 nM T20251 CGP38T 45482687 IC50 = 7543.86 nM T20251 CHV1Q5 45482688 IC50 = 323333.33 nM T20251 CK2G6S 45482693 IC50 = 6666.67 nM T20251 C9L4FG 45482694 IC50 = 1111.11 nM T20251 CEY8O1 45482699 IC50 = 989.01 nM T20251 C7W0DZ 45482705 IC50 = 19411.76 nM T20251 CP2ZT9 45482708 IC50 = 1111.11 nM T20251 CRL9I4 45482709 IC50 = 8181.82 nM T20251 C9UE0Y 45482713 IC50 = 101.01 nM T20251 C3P5TG 45482727 IC50 = 40000 nM T20251 CZM43G 45482728 IC50 = 190000 nM T20251 CB8E2S 45482734 IC50 = 196000 nM T20251 CDM1L4 45482735 IC50 = 80000 nM T20251 CEM05T 45482739 IC50 = 43000 nM T20251 C2LU1K 45482740 IC50 = 140000 nM T20251 CHQ4M5 45482745 IC50 = 23333.33 nM T20251 CJ3X8T 45482746 IC50 = 190000 nM T20251 C3NC6W 45482751 IC50 = 1235.96 nM T20251 CX9RG6 45482752 IC50 = 40000 nM T20251 C28XSF 45482753 IC50 = 8518.52 nM T20251 CZLA81 45482756 IC50 = 9607.84 nM T20251 CIH4Z3 45482757 IC50 = 6393.44 nM T20251 C4EIV8 45482763 IC50 = 132857.14 nM T20251 CE0H4S 45482770 IC50 = 1764.71 nM T20251 CLKA86 45482775 IC50 = 101.01 nM T20251 C2ED8W 45482783 IC50 = 309.28 nM T20251 C0CHF4 45482789 IC50 > 30000 nM T20251 C8YIM9 45483679 IC50 = 411 nM T20251 CE4LA5 45483880 IC50 = 11220.18 nM T20251 CX12QY 45483901 IC50 = 3467.37 nM T20251 C0TED2 45483913 IC50 = 4168.69 nM T20251 CMQ17N 45484111 IC50 = 5600 nM T20251 C5YT2N 45484113 IC50 = 4400 nM T20251 C85XBW 45484115 IC50 = 12200 nM T20251 C9D6SC 45484116 IC50 = 33000 nM T20251 CO42HZ 45484117 IC50 = 28300 nM T20251 CC8X7E 45485452 Ki = 431 nM T20251 C3AT2W 45485462 IC50 > 100000 nM T20251 CSQ1J5 45487336 IC50 > 10000 nM T20251 C3QU2C 45487384 IC50 = 5100 nM T20251 C24WVU 45487513 IC50 = 6309.57 nM T20251 CMX27T 45487640 IC50 = 530 nM T20251 C5NO1K 45487641 IC50 > 10000 nM T20251 CR10DI 45487647 IC50 = 17 nM T20251 CS17WK 45487652 IC50 = 24 nM T20251 CAQ2D8 45487653 IC50 = 3670 nM T20251 C3A7QW 45487657 IC50 = 23 nM T20251 CB9K2G 45487660 IC50 = 25 nM T20251 CJ8R3S 45487668 IC50 = 250 nM T20251 CN1V0Y 45487671 IC50 = 140 nM T20251 CWH0O7 45487673 IC50 = 520 nM T20251 CCZR81 45487674 IC50 = 1790 nM T20251 C80FMT 45487762 Ki = 4200 nM T20251 CR0X4I 45487870 Ki = 1600 nM T20251 CL32NJ 45488686 IC50 = 19000 nM T20251 C32YDN 46175430 IC50 = 50118.72 nM T20251 CH5Y4W 46175432 IC50 > 100000 nM T20251 C6MI2B 46175433 IC50 = 36000 nM T20251 CZ8SI1 46175518 IC50 = 19952.62 nM T20251 CR9J1S 46175520 IC50 = 62000 nM T20251 CZKB10 46175521 IC50 = 10000 nM T20251 CA6G8I 46175610 IC50 = 50118.72 nM T20251 C2L3HT 46175611 IC50 > 100000 nM T20251 C7CK6V 46178246 IC50 = 4800 nM T20251 CP12AF 46179404 IC50 > 30000 nM T20251 CS8TU3 46179405 IC50 > 30000 nM T20251 CR0I3A 46180744 IC50 = 8700 nM T20251 C7W2LJ 46180746 IC50 = 2200 nM T20251 CL7F3D 46187355 IC50 > 30000 nM T20251 CNDF17 46187356 IC50 > 80000 nM T20251 CZ8N7D 46197576 IC50 = 27600 nM T20251 CF9QB5 46197577 IC50 = 13400 nM T20251 CMK3H7 46197578 IC50 = 9100 nM T20251 C7IGB2 46197685 IC50 = 29300 nM T20251 C9T7FD 46197686 IC50 = 28400 nM T20251 C8IQ5Z 46197687 IC50 = 13500 nM T20251 CJZ3X6 46197795 IC50 = 19300 nM T20251 C7Z6JK 46197796 IC50 = 30000 nM T20251 C9Z6UF 46197797 IC50 = 9900 nM T20251 CFKV19 46197898 IC50 = 15300 nM T20251 CYAI40 46198106 IC50 = 20000 nM T20251 CTI0F8 46198107 IC50 > 80000 nM T20251 CJ9OY8 46198108 IC50 = 10000 nM T20251 CI9QH8 46198109 IC50 > 80000 nM T20251 CU3VQ1 46198110 IC50 = 7300 nM T20251 C2P9ST 46198216 IC50 = 38000 nM T20251 CSEL57 46198325 IC50 = 53000 nM T20251 C2VIF3 46198326 IC50 = 8600 nM T20251 C6JWH5 46198327 IC50 = 25900 nM T20251 C13RUW 46198329 IC50 = 26000 nM T20251 CRLM46 46201983 IC50 = 1000 nM T20251 C7VR2G 46202081 IC50 = 3500 nM T20251 C56SZE 46202415 IC50 = 7200 nM T20251 C38LWQ 46202743 IC50 = 3800 nM T20251 C4A5NH 46203391 IC50 = 2100 nM T20251 CFYP54 46203897 IC50 < 400 nM T20251 CBQ31T 46205018 IC50 > 100000 nM T20251 C9L4KT 46205341 IC50 > 333000 nM T20251 C4OK3I 46205343 IC50 > 333000 nM T20251 C1A5VL 46205345 IC50 > 333000 nM T20251 CX8OB9 46205674 IC50 = 174000 nM T20251 C9MPG6 46205967 IC50 = 5700 nM T20251 CNVX45 46205968 IC50 = 3100 nM T20251 CL41FE 46206000 IC50 > 333000 nM T20251 CR9A5G 46206291 IC50 = 16000 nM T20251 C9B1CG 46206292 IC50 = 7900 nM T20251 CSX8P1 46206294 IC50 = 1600 nM T20251 CD0R7T 46206296 IC50 = 500 nM T20251 C3X4KZ 46206324 IC50 > 333000 nM T20251 CR1X0F 46206642 IC50 = 11000 nM T20251 C8JYQ3 46206643 IC50 = 6400 nM T20251 C0R1YT 46206645 IC50 = 1700 nM T20251 CH8Y7D 46206977 IC50 = 2200 nM T20251 C9FI2Z 46208126 IC50 = 13000 nM T20251 CE45XW 46208354 IC50 = 360 nM T20251 CUHB49 46208355 IC50 = 7700 nM T20251 CW38GO 46208357 IC50 = 17000 nM T20251 C43COY 46208358 IC50 = 8100 nM T20251 CE4Q7D 46208596 IC50 = 4800 nM T20251 CM9UN7 46208601 IC50 > 100000 nM T20251 CMG47W 46208633 IC50 = 7500 nM T20251 CLUF01 46208857 IC50 = 6400 nM T20251 CO3Y7Q 46208858 IC50 = 12000 nM T20251 CH7JB4 46209051 IC50 > 100000 nM T20251 C0SNL2 46209134 IC50 = 21000 nM T20251 C5KFD3 46212800 IC50 > 33000 nM T20251 CB04XO 46212809 IC50 > 33000 nM T20251 C6U0CX 46212866 IC50 > 33000 nM T20251 CU6X8G 46213054 Ki = 690 nM T20251 CL51NF 46216732 Ki = 2560 nM T20251 CZJL95 46216733 Ki = 4910 nM T20251 C8BN4H 46216788 IC50 = 11000 nM T20251 C57OFD 46216800 IC50 = 12000 nM T20251 C3JUH5 46216812 IC50 = 8000 nM T20251 CPI8M7 46224242 IC50 = 5800 nM T20251 C0TYK4 46224262 IC50 = 8900 nM T20251 C26LPQ 46225987 IC50 = 9500 nM T20251 CHO7G1 46226010 IC50 = 15800 nM T20251 CDS61T 46226025 IC50 = 40100 nM T20251 CARU41 46226027 IC50 = 135000 nM T20251 CA2L5H 46227092 Ki = 4620 nM T20251 CLS58Y 46227093 Ki = 300 nM T20251 CH5VD2 46227102 Ki = 3000 nM T20251 C1DO4U 46230960 Ki = 3310 nM T20251 C59XOB 46230961 Ki = 1650 nM T20251 C9EGU1 46230962 Ki > 4760 nM T20251 C2FVA8 46231075 IC50 = 1540 nM T20251 CA3R5W 46231076 IC50 = 1720 nM T20251 CSZ2F6 46231077 Ki = 2110 nM T20251 CVL6C0 46231146 Ki > 5190 nM T20251 C8W4VL 46231147 Ki = 4530 nM T20251 CRTO63 46231148 Ki = 177 nM T20251 CZ6C0S 46231149 Ki = 3810 nM T20251 C8RP5H 46232900 IC50 > 90000 nM T20251 C7OB2G 46235733 IC50 = 6400 nM T20251 CZK5E9 46238536 IC50 = 7500 nM T20251 CY2A9C 46240380 IC50 = 22500 nM T20251 CIG71O 46240381 IC50 > 50000 nM T20251 CFY3L5 46240481 IC50 = 43800 nM T20251 CPHB87 46240482 IC50 = 32000 nM T20251 C8R1QX 46240484 IC50 = 28000 nM T20251 CR0NX3 46240582 IC50 = 15000 nM T20251 CF9O5C 46240584 IC50 = 6200 nM T20251 CV2X5E 46240585 IC50 > 50000 nM T20251 CD1M3J 46240687 IC50 = 6000 nM T20251 C63QWF 46240785 IC50 > 50000 nM T20251 C3YU2T 46240895 IC50 = 24000 nM T20251 CEH6U9 46241010 IC50 = 28000 nM T20251 C43MLP 46241011 IC50 > 50000 nM T20251 CJ7L3Z 46241120 IC50 = 27000 nM T20251 C7PVU1 46241121 IC50 > 50000 nM T20251 CDZ3V6 46241509 IC50 = 37000 nM T20251 CH8F5U 46241608 IC50 = 11200 nM T20251 CD1H3B 46241609 IC50 = 25000 nM T20251 CXJ7C5 46241610 IC50 = 5500 nM T20251 C35CXM 46241611 IC50 = 17500 nM T20251 C5Y8ZT 46241717 IC50 = 14500 nM T20251 C8EX9T 46241718 IC50 = 9800 nM T20251 CZK4H8 46241719 IC50 = 10000 nM T20251 CK9H6B 46241720 IC50 = 12500 nM T20251 CA05ZH 46241826 IC50 = 35000 nM T20251 C3LD6V 46241827 IC50 = 21600 nM T20251 CRJD47 46241829 IC50 = 35000 nM T20251 CL7C2K 46244173 IC50 > 100000 nM T20251 C2NH0A 46244259 IC50 > 33000 nM T20251 CVJM38 46244260 IC50 > 33000 nM T20251 C31PAF 46700737 IC50 = 17000 nM T20251 CJ2D3O 46701015 IC50 = 5280 nM T20251 CM04ZI 46701016 IC50 = 5640 nM T20251 C0JWP5 46701017 IC50 = 5430 nM T20251 C5H0MJ 46701086 IC50 = 6480 nM T20251 C9HWI7 46701087 IC50 = 3640 nM T20251 CVE5O1 46701088 IC50 = 2320 nM T20251 C1VPM0 46701089 IC50 = 4140 nM T20251 CQ8B6R 46701090 IC50 = 4330 nM T20251 C6C0FS 46701091 IC50 = 4730 nM T20251 C2ILJ9 46701790 Ki = 1258.93 nM T20251 C2SOY1 46785920 IC50 > 30000 nM T20251 CCJ08W 46830055 IC50 = 39900 nM T20251 CC68WI 46830289 IC50 = 2000 nM T20251 CC3UF9 46830325 IC50 = 5100 nM T20251 C5TC2S 46830335 IC50 > 10000 nM T20251 C1K7FL 46830336 IC50 > 10000 nM T20251 C2ZGO0 46830791 IC50 = 8000 nM T20251 CL7XJ8 46831392 IC50 = 13000 nM T20251 CEV89K 46831395 IC50 = 20000 nM T20251 CICY27 46833073 IC50 = 4100 nM T20251 C6G1DY 46833075 IC50 = 900 nM T20251 C7MU0O 46835136 IC50 = 500 nM T20251 C9CR0E 46835922 IC50 = 18000 nM T20251 CGS4F2 46836713 IC50 = 30000 nM T20251 C0GY1V 46837247 IC50 > 40000 nM T20251 CQ41PO 46837248 IC50 > 40000 nM T20251 CN1EK8 46837249 IC50 > 40000 nM T20251 C6IXU7 46837365 IC50 = 10000 nM T20251 C0M8AW 46839029 IC50 = 2000 nM T20251 C1ZDW9 46839030 IC50 = 3000 nM T20251 C21ILB 46839164 IC50 = 1200 nM T20251 C1OIG5 46839165 IC50 = 10000 nM T20251 C9S4IH 46839298 IC50 = 6900 nM T20251 C1EPB3 46839300 IC50 = 20000 nM T20251 C1N4KX 46842383 IC50 > 10000 nM T20251 CIM53K 46847263 IC50 = 13800 nM T20251 CO7G8Z 46851863 IC50 = 4040 nM T20251 C4S6YJ 46853439 IC50 = 170 nM T20251 CO31WX 46861576 IC50 = 8500 nM T20251 CC5IO9 46861756 IC50 > 10000 nM T20251 C19ZCY 46861765 IC50 = 4970 nM T20251 CP6DN0 46861858 Ki = 5291 nM T20251 C5VOF1 46861859 Ki = 1373 nM T20251 CW1FS9 46861860 Ki > 10000 nM T20251 C2QH7O 46865650 Ki > 3000 nM T20251 CC2O9R 46865656 IC50 = 19952.62 nM T20251 CQN2H4 46865774 IC50 > 80000 nM T20251 CPV2L4 46865775 IC50 = 30000 nM T20251 CC5KR7 46865978 Ki > 3000 nM T20251 CC7DG3 46866398 IC50 = 1100 nM T20251 CO3P0J 46866604 IC50 > 30000 nM T20251 CS9LD5 46867516 IC50 > 30000 nM T20251 C1XGZ8 46867925 IC50 > 30000 nM T20251 CZQ57K 46868086 IC50 = 2300 nM T20251 C9NGO7 46869046 IC50 = 18000 nM T20251 C8BT1F 46869326 IC50 = 12000 nM T20251 C97JEP 46871671 IC50 = 120 nM T20251 C8JZ2A 46871848 IC50 > 30000 nM T20251 CLS29B 46872626 IC50 = 77000 nM T20251 CFZ75O 46880148 IC50 > 30000 nM T20251 C0PXY7 46880628 IC50 > 10000 nM T20251 C2MC4K 46881463 IC50 = 7943.28 nM T20251 CSQ4C9 46881468 IC50 = 15848.93 nM T20251 C4BH9E 46882458 IC50 = 2511.89 nM T20251 CAH31I 46882578 IC50 = 180 nM T20251 CMS27C 46882857 IC50 > 40000 nM T20251 CM45ZP 46882858 IC50 = 7920 nM T20251 C3IGF1 46882859 IC50 = 19800 nM T20251 CHLZ97 46882860 IC50 > 10000 nM T20251 C4B8EX 46882909 IC50 = 4120 nM T20251 CFY95C 46882910 IC50 = 52400 nM T20251 C0SQX2 46882912 IC50 > 10000 nM T20251 CJ82WI 46882913 IC50 > 10000 nM T20251 CM5Z4G 46882938 IC50 = 12900 nM T20251 C60YMF 46883462 IC50 > 20000 nM T20251 C7J6GU 46883497 IC50 > 18600 nM T20251 C3F5AS 46883498 IC50 = 7140 nM T20251 CRSE34 46883499 IC50 = 16800 nM T20251 C0CX3O 46883500 IC50 = 7740 nM T20251 C15KEH 46883819 IC50 = 12700 nM T20251 C3J5IG 46883820 IC50 = 7880 nM T20251 CGKP83 46883876 IC50 = 3810 nM T20251 CJ39QM 46883878 IC50 = 384 nM T20251 CXIM81 46883917 IC50 = 12000 nM T20251 C3OBL5 46883918 IC50 = 2310 nM T20251 CR6FO1 46883919 IC50 = 13800 nM T20251 CW6A9I 46884062 Ki > 5000 nM T20251 C04JMO 46884063 Ki = 0.73 nM T20251 CR1Z8E 46884119 Ki > 5000 nM T20251 CR0CQ9 46884120 IC50 = 3000 nM T20251 C9OYT5 46884152 IC50 = 330 nM T20251 CCI32B 46884153 Ki > 5000 nM T20251 C2JQE7 46884154 Ki > 5000 nM T20251 C20HET 46884155 Ki > 5000 nM T20251 C0HYN3 46884200 IC50 = 1500 nM T20251 CM6A8S 46884201 IC50 = 1700 nM T20251 CW94IK 46884202 Ki > 5000 nM T20251 C3QT0U 46884239 Ki > 5000 nM T20251 CYC64I 46884402 IC50 = 61 nM T20251 CF7HD6 46884426 IC50 = 178 nM T20251 C9M4RX 46884427 IC50 = 188 nM T20251 CT9K2R 46884428 IC50 = 202 nM T20251 CWK75U 46884462 IC50 = 6650 nM T20251 C82IYB 46884463 IC50 = 9190 nM T20251 COPQ16 46884600 Ki > 3000 nM T20251 C85MOA 46884637 Ki > 3000 nM T20251 C36NKV 46884638 Ki > 3000 nM T20251 CQ84IF 46884639 Ki > 3000 nM T20251 CZGS15 46884640 Ki > 3000 nM T20251 CZ72SW 46884641 Ki > 3000 nM T20251 CA3Z6G 46884666 Ki > 3000 nM T20251 C8DBY0 46884667 IC50 = 1900 nM T20251 CU3BG6 46884668 IC50 = 520 nM T20251 CPG14Q 46884669 IC50 = 2100 nM T20251 C7R9AK 46884670 IC50 = 110 nM T20251 C64KNW 46884698 IC50 = 230 nM T20251 C0ASK4 46884699 IC50 = 360 nM T20251 CYNU85 46884731 Ki > 3000 nM T20251 CJ6O8D 46884732 Ki > 3000 nM T20251 C9QT7G 46884733 Ki > 3000 nM T20251 CL6Z7Q 46884734 IC50 = 1800 nM T20251 C6PRX8 46884735 Ki = 1200 nM T20251 CWK8I4 46884736 IC50 = 620 nM T20251 CB8GE1 46884818 IC50 > 10000 nM T20251 C4MQ0A 46884856 IC50 = 10000 nM T20251 CCNT25 46884898 IC50 > 10000 nM T20251 C3MSG2 46885027 IC50 > 10000 nM T20251 CB7XI0 46885213 IC50 > 10000 nM T20251 CD3E4C 46885323 Ki = 6.65 nM T20251 CNW43Y 46885367 Ki > 9.17 nM T20251 CV23JL 46885415 Ki = 5.87 nM T20251 CHPS01 46885417 Ki > 5.27 nM T20251 C4SVE1 46885480 Ki = 4.65 nM T20251 C5QI7J 46885481 Ki = 5.07 nM T20251 COU5X2 46885482 Ki > 10 nM T20251 C1TXI0 46885514 IC50 > 60000 nM T20251 CS90MN 46885524 Ki > 10 nM T20251 CQ94VM 46885526 Ki > 10 nM T20251 C90ABZ 46885558 Ki > 10 nM T20251 CKF74T 46885587 IC50 > 60000 nM T20251 CKH5W7 46885611 IC50 = 2300 nM T20251 C0Y9NF 46885711 Ki > 10 nM T20251 C3O5BR 46885712 Ki = 7.91 nM T20251 CK8D6G 46885760 Ki = 5 nM T20251 CY30PG 46885815 Ki = 5.84 nM T20251 CFC5L1 46885972 Ki > 7.88 nM T20251 CF8N0U 46886536 IC50 = 3000 nM T20251 CZ59HO 46886537 IC50 > 80000 nM T20251 C28IHA 46886538 IC50 = 4000 nM T20251 C0UDN9 46886539 IC50 = 22000 nM T20251 CO2PM3 46887855 IC50 = 1320 nM T20251 C8EOA7 46887961 IC50 = 3000 nM T20251 C0XR8B 46887962 IC50 = 7800 nM T20251 CE4X6C 46887963 IC50 = 2000 nM T20251 CVB6C0 46887993 IC50 = 7200 nM T20251 C0U3CX 46887994 IC50 > 10000 nM T20251 CG8I9K 46887995 IC50 = 2900 nM T20251 CVY2T4 46888365 IC50 = 2000 nM T20251 CO7M5J 46888366 IC50 = 4600 nM T20251 CLS1G3 46888367 IC50 = 630 nM T20251 CGD6T5 46888386 IC50 > 30000 nM T20251 C13SVO 46888387 IC50 = 540 nM T20251 C9G2HI 46888388 IC50 = 2660 nM T20251 C5D2CK 46888389 IC50 > 30000 nM T20251 CAE10V 46888443 IC50 > 10000 nM T20251 C9QO6J 46888468 IC50 > 10000 nM T20251 C6DB3K 46888487 IC50 > 10000 nM T20251 CM76UZ 46888550 IC50 > 10000 nM T20251 CQ5B2F 46888578 IC50 = 2800 nM T20251 CDUM26 46888645 IC50 = 300 nM T20251 CTN16E 46888688 IC50 = 600 nM T20251 C4SX5W 46888719 IC50 = 80 nM T20251 CT8E9F 46888720 IC50 > 30000 nM T20251 CP75RD 46888721 IC50 > 30000 nM T20251 C9Z2CO 46888748 IC50 = 1200 nM T20251 CR7HN9 46888749 IC50 = 5300 nM T20251 C06HUF 46888750 IC50 = 8700 nM T20251 CEMZ98 46888775 IC50 > 30000 nM T20251 CYT7P0 46888776 IC50 = 380 nM T20251 CJDH10 46888777 IC50 = 1100 nM T20251 CM6S8Z 46888778 IC50 = 1600 nM T20251 CZBL19 46888785 Ki > 5000 nM T20251 CK3B2R 46888786 Ki = 1262 nM T20251 C46QKX 46888787 Ki > 10000 nM T20251 CJS87P 46888788 Ki > 10000 nM T20251 C98ROS 46888789 Ki = 638 nM T20251 C9RXL8 46888825 Ki = 926 nM T20251 CHN7W1 46888826 Ki = 2649 nM T20251 C46PXH 46888827 Ki = 1840 nM T20251 CR42EN 46888828 Ki > 10000 nM T20251 C3B2QN 46888853 Ki > 10000 nM T20251 C94FRI 46888854 Ki > 3000 nM T20251 C30FVT 46888855 Ki = 1183 nM T20251 C4Q2MA 46888856 Ki > 3000 nM T20251 CJK1Z5 46888857 IC50 = 720 nM T20251 C4U3CN 46888882 Ki = 6515 nM T20251 C61GZW 46888883 Ki > 10000 nM T20251 C6KOP3 46888884 Ki > 10000 nM T20251 C4AFL7 46888885 Ki = 10336 nM T20251 CC8G6T 46888886 Ki > 10000 nM T20251 C3V4ZN 46888887 IC50 = 2100 nM T20251 CX92WH 46889257 IC50 = 492 nM T20251 C01DMO 46889258 IC50 = 233 nM T20251 C2CI9O 46889753 IC50 = 7500 nM T20251 C3J5IQ 46889754 IC50 = 35000 nM T20251 CX18GT 46889932 IC50 = 3000 nM T20251 CM12LB 46889933 IC50 = 2300 nM T20251 CL51ME 46890090 Ki = 440 nM T20251 C2XCK5 46890181 Ki = 1200 nM T20251 CTS04G 46890283 Ki = 4500 nM T20251 CV8C4E 46890347 Ki = 5600 nM T20251 CH56AN 46890391 IC50 = 6370 nM T20251 CPDX34 46890392 IC50 = 6400 nM T20251 C0YGP2 46890393 IC50 = 2960 nM T20251 C61INJ 46890394 IC50 = 21400 nM T20251 C4XLV0 46890430 Ki = 5600 nM T20251 CI14SE 46890441 IC50 = 20800 nM T20251 CP4GD3 46890442 IC50 = 8550 nM T20251 CQI2Y8 46890443 IC50 = 10400 nM T20251 CZ2MG7 46890444 IC50 = 40100 nM T20251 CP6A8K 46890445 IC50 > 22500 nM T20251 CD5J8B 46890446 IC50 = 16000 nM T20251 C4IK6F 46890475 Ki = 2100 nM T20251 CK08VN 46890476 Ki = 6200 nM T20251 CYK9D2 46890489 IC50 = 6500 nM T20251 CCR04L 46890490 IC50 = 8240 nM T20251 CT4O9M 46890491 IC50 = 9120 nM T20251 CGPM19 46890493 IC50 = 6110 nM T20251 CM56CG 46890523 Ki = 6900 nM T20251 C2K4HZ 46890562 Ki = 780 nM T20251 C89ZNE 46890564 Ki = 54000 nM T20251 CT4Q8R 46890603 Ki = 1700 nM T20251 C6XPD3 46890638 Ki = 4400 nM T20251 CQLS54 46890639 Ki = 4200 nM T20251 CP7ZS3 46890640 Ki = 1500 nM T20251 CU3O0K 46890688 Ki = 10000 nM T20251 CZ0A7U 46890769 Ki = 5.3 nM T20251 C1AK8C 46890770 Ki = 1.2 nM T20251 CB6T3M 46890771 Ki > 65 nM T20251 CP8FW2 46890772 Ki = 14 nM T20251 CX7I3Y 46890773 Ki = 1.9 nM T20251 C3MPJ7 46890808 Ki > 9000 nM T20251 C2I9CM 46890824 Ki > 51 nM T20251 C6RB1V 46890825 Ki = 9 nM T20251 C5JT1D 46890826 Ki = 22 nM T20251 CC0E7P 46890827 Ki = 1.3 nM T20251 CT6UY7 46890828 Ki = 0.56 nM T20251 C9QFU5 46890891 Ki > 35 nM T20251 CS74RA 46890892 Ki = 4.3 nM T20251 CNQ26O 46890893 Ki = 1.85 nM T20251 CZQ25U 46890894 Ki = 13 nM T20251 CJ8YV7 46890895 Ki = 10 nM T20251 CWDG43 46890952 Ki = 2.7 nM T20251 CIC32L 46890953 Ki = 0.55 nM T20251 C4ZYM8 46890954 Ki = 46 nM T20251 C0P4GM 46890955 Ki = 11 nM T20251 CK94BQ 46890956 Ki = 2 nM T20251 CEW98A 46891012 Ki = 32 nM T20251 C3CPE9 46891013 Ki = 2.9 nM T20251 C51IBN 46891527 Ki = 8.8 nM T20251 CQ34CV 46891528 Ki = 1.8 nM T20251 CH91DV 46891529 Ki > 55 nM T20251 C7LS0J 46891530 Ki = 21 nM T20251 CCE34G 46891585 Ki = 2.2 nM T20251 CMJ93X 46891586 Ki > 57 nM T20251 CHGA57 46891587 Ki = 12 nM T20251 C2FOK8 46891588 Ki = 12 nM T20251 C4ZXM7 46891589 Ki = 26 nM T20251 CZ7C1J 46893145 Ki = 2900 nM T20251 CS8XC4 46893453 IC50 = 29512.09 nM T20251 C5F1CH 46893542 IC50 > 100000 nM T20251 C90NYX 46896338 IC50 = 10000 nM T20251 CC9FZ0 46898063 IC50 = 10500 nM T20251 C1JSH9 46899637 Ki = 199.53 nM T20251 C3MSL0 46899638 Ki = 501.19 nM T20251 CV3LP2 46899639 Ki = 1258.93 nM T20251 CGHZ15 46899640 Ki = 1000 nM T20251 CN9FC3 46900150 Ki = 1584.89 nM T20251 C40ZJO 46900451 Ki = 398.11 nM T20251 CNC02A 46900453 Ki = 398.11 nM T20251 CTCH14 46900455 Ki = 25.12 nM T20251 CP41AQ 46900457 Ki = 1000 nM T20251 CR3L4I 46900459 Ki = 12589.25 nM T20251 CK17PA 46900606 Ki = 2511.89 nM T20251 CQ2K1C 46900608 Ki = 501.19 nM T20251 C5ZT1B 46900610 Ki = 7943.28 nM T20251 C1NAX4 46900612 Ki = 6309.57 nM T20251 CT0SQ2 46900614 Ki = 2511.89 nM T20251 CXD9S3 46900776 Ki = 3981.07 nM T20251 C8I7SJ 46900778 Ki = 1000 nM T20251 C7QDM9 46900782 Ki = 2511.89 nM T20251 C15FMY 46900954 Ki = 630.96 nM T20251 C8W1FU 46900956 Ki = 501.19 nM T20251 CH35BV 46900958 Ki = 199.53 nM T20251 C7T2GX 46909057 IC50 = 37000 nM T20251 CZ46AH 46911015 IC50 = 1690 nM T20251 C3JCB1 46911060 IC50 > 100000 nM T20251 CA2JU7 46911115 IC50 = 4000 nM T20251 C73VYX 46911116 IC50 = 6000 nM T20251 C1MEW3 46911124 IC50 > 300000 nM T20251 C4DTN2 46911175 IC50 = 5900 nM T20251 C5XAF7 46912235 IC50 = 9000 nM T20251 CE7KZ8 46914881 IC50 = 170 nM T20251 CI0Y4F 46914882 IC50 > 30000 nM T20251 C8HWO7 46914883 IC50 > 30000 nM T20251 C6FN4G 46914884 IC50 > 30000 nM T20251 CY3O2C 46915043 IC50 = 29 nM T20251 CR5OZ8 46916382 IC50 = 2000 nM T20251 C0HZ4C 46916514 IC50 > 10000 nM T20251 CDBM59 46916519 IC50 > 10000 nM T20251 CW6Y2D 46916520 IC50 > 10000 nM T20251 CK9E8N 46927116 IC50 = 10000 nM T20251 C82HXR 46927117 IC50 = 2800 nM T20251 C8GAI9 46927903 IC50 = 1995.26 nM T20251 C3D7FL 46931619 Ki = 1100 nM T20251 CW3L9K 46931735 IC50 = 4200 nM T20251 CKO76R 46931815 IC50 = 1000 nM T20251 C3M4LT 46931848 IC50 = 9800 nM T20251 C9EG4R 46931852 IC50 = 2800 nM T20251 CB84WK 46931947 IC50 = 10300 nM T20251 CJMS30 46931948 IC50 = 3200 nM T20251 C2M1KO 46932044 Ki = 1700 nM T20251 C3QLC4 46932045 Ki = 2800 nM T20251 CC91MK 46932046 Ki = 3400 nM T20251 CQ91FA 46932047 Ki = 3900 nM T20251 CYCF24 46932049 Ki = 6200 nM T20251 C3O4MA 46932136 Ki = 6000 nM T20251 CF9YV2 46932138 Ki = 4200 nM T20251 COL7J6 46932139 Ki = 10500 nM T20251 CSMK50 46932141 Ki = 3300 nM T20251 C29RXO 46932234 Ki = 21200 nM T20251 CC0F4D 46932235 Ki = 13700 nM T20251 C8QB4Z 46932237 Ki = 9800 nM T20251 CG2J9V 46932512 Ki = 15300 nM T20251 C2VZ7Q 46932514 Ki = 19500 nM T20251 C4PW3A 46932704 Ki > 60000 nM T20251 C82QKP 46932796 IC50 = 4800 nM T20251 COY21M 46935743 IC50 = 69000 nM T20251 CU90MG 46938037 IC50 > 1000000000 nM T20251 CX2U5I 46938097 IC50 > 1000000000 nM T20251 C47QBL 46938101 IC50 > 1000000000 nM T20251 CV28ZU 46944853 IC50 = 6200 nM T20251 CT9P5G 46944854 IC50 = 8200 nM T20251 CWH4K6 46944855 IC50 = 23000 nM T20251 CC3O0S 46945254 IC50 = 44000 nM T20251 C1UB8E 46945255 IC50 = 37000 nM T20251 C4RZG5 46945857 IC50 = 12000 nM T20251 CAK5J0 46946058 IC50 = 9800 nM T20251 CY09UB 46946452 IC50 = 2400 nM T20251 C6J4TV 46946859 Ki = 1850 nM T20251 CFH87K 46947816 IC50 = 10000 nM T20251 CVEF51 49763568 IC50 = 2800 nM T20251 C43LAE 49763569 IC50 = 2800 nM T20251 CI6AR9 49763571 IC50 = 4000 nM T20251 C78ICP 49763574 IC50 = 3300 nM T20251 C65RMG 49763575 IC50 = 6200 nM T20251 CQLN97 49763682 IC50 = 3000 nM T20251 CY5ME3 49763685 IC50 = 1300 nM T20251 C0ADU9 49763686 IC50 = 23000 nM T20251 C1GVM0 49763804 IC50 = 7900 nM T20251 C94ARN 49763931 IC50 = 2500 nM T20251 C68SFM 49764196 IC50 = 13500 nM T20251 CSW83Q 49764322 IC50 = 8900 nM T20251 C1Z0UD 49764446 IC50 = 25000 nM T20251 C5AD0E 49764447 IC50 = 4100 nM T20251 C20WNR 49764700 IC50 = 2800 nM T20251 CIZ86P 49764701 IC50 = 1500 nM T20251 CABL63 49765080 IC50 = 2 nM T20251 CIXN24 49767138 IC50 = 1600 nM T20251 CR13SJ 49767146 IC50 = 4300 nM T20251 CZWN54 49767224 IC50 = 6900 nM T20251 CDM18G 49768863 IC50 = 4230 nM T20251 CWU2R3 49773361 IC50 = 12400 nM T20251 CYWX19 49780808 IC50 = 7943.28 nM T20251 C9RI3L 49780809 IC50 = 251.19 nM T20251 C39KWP 49781039 IC50 = 2511.89 nM T20251 C9O2RB 49781040 IC50 = 630.96 nM T20251 C7T3KS 49781255 IC50 = 316.23 nM T20251 CYL65E 49781476 IC50 = 158.49 nM T20251 CFQN89 49781477 IC50 = 501.19 nM T20251 CL82ES 49781478 IC50 = 501.19 nM T20251 CAFW31 49783666 IC50 = 26000 nM T20251 CNI1P6 49783903 IC50 > 33000 nM T20251 CGF65B 49783985 IC50 > 33000 nM T20251 CZ7A9E 49796933 IC50 = 9700 nM T20251 C5RF0Y 49796938 IC50 > 90000 nM T20251 CE0C3Y 49796939 IC50 = 79000 nM T20251 CI25XP 49796945 IC50 = 870 nM T20251 C8WYA5 49796953 IC50 = 76000 nM T20251 CQH86V 49796955 IC50 > 100000 nM T20251 CBMV50 49796972 Ki = 1100 nM T20251 CX74RG 49796999 IC50 = 4600 nM T20251 C7B5DY 49797060 IC50 = 59000 nM T20251 CA2U4Y 49797089 IC50 > 100000 nM T20251 CBS36X 49797110 IC50 > 100000 nM T20251 C0STP5 49797111 IC50 > 100000 nM T20251 C2OI0Y 49797114 IC50 = 8300 nM T20251 CW20FJ 49797115 IC50 > 100000 nM T20251 CY1OJ5 49797177 Ki > 50000 nM T20251 C25ZSD 49797191 IC50 = 36700 nM T20251 C6ZGL5 49797198 IC50 > 100000 nM T20251 CON0A6 49797232 IC50 = 26100 nM T20251 CA4E8M 49797242 IC50 = 9900 nM T20251 C37MDP 49797244 IC50 = 8100 nM T20251 CUMH43 49797248 IC50 = 33200 nM T20251 C93VJO 49797347 IC50 > 90000 nM T20251 C1Z8HB 49797353 IC50 = 49000 nM T20251 CTYO37 49797358 IC50 > 90000 nM T20251 C1K4FR 49797359 IC50 = 78000 nM T20251 CA3Q2W 49797361 IC50 > 90000 nM T20251 CNMF62 49797362 IC50 = 39000 nM T20251 C76KMB 49797451 IC50 = 37000 nM T20251 CU72EZ 49797596 IC50 = 17000 nM T20251 C6DJX7 49797605 IC50 = 38000 nM T20251 CK3ZI1 49797607 IC50 = 2500 nM T20251 CV6I0O 49797630 IC50 = 7500 nM T20251 CQVG17 49798349 IC50 = 7943.28 nM T20251 C62VRQ 49798437 IC50 > 63095.73 nM T20251 CY90CD 49798461 IC50 > 31622.78 nM T20251 C5I1HQ 49798777 IC50 = 20000 nM T20251 C02EUQ 49800098 IC50 = 8130 nM T20251 CM75QU 49801042 IC50 = 2400 nM T20251 C8LFB9 49801043 IC50 = 9000 nM T20251 C8IYR7 49801044 IC50 = 3500 nM T20251 C8A0LD 49801837 IC50 = 28000 nM T20251 CP91TS 49802222 IC50 = 16000 nM T20251 CIFZ02 49803320 IC50 = 28000 nM T20251 CEP3B7 49803607 IC50 > 30000 nM T20251 C1BLY0 49804185 IC50 = 40000 nM T20251 C97LZE 49804478 IC50 = 5200 nM T20251 C2IGB7 49804777 IC50 = 2200 nM T20251 C73PSQ 49805872 IC50 > 3000 nM T20251 CML8Z5 49805873 IC50 > 10000 nM T20251 C41TPM 49806128 IC50 > 3000 nM T20251 C4O0QK 49821278 Ki = 13000 nM T20251 CDAB96 49836026 IC50 = 1995.26 nM T20251 CI8FT3 49836033 IC50 > 33000 nM T20251 CO20JE 49836187 IC50 > 63095.73 nM T20251 CT7CV0 49836295 IC50 > 39810.72 nM T20251 CYJW87 49836299 IC50 > 63095.73 nM T20251 C8E6WA 49836410 IC50 > 39810.72 nM T20251 CNM9X8 49836528 IC50 > 39810.72 nM T20251 COK75S 49836633 IC50 > 50118.72 nM T20251 CB71TA 49837867 IC50 = 700 nM T20251 CZQC64 49837869 IC50 > 20000 nM T20251 CVNA15 49837870 IC50 > 20000 nM T20251 C9L3XR 49838879 IC50 > 160000 nM T20251 CL64TH 49842175 IC50 > 10000 nM T20251 C3T6NH 49843555 Ki = 3700 nM T20251 CU63QR 49847377 IC50 = 22000 nM T20251 CZT4I8 49847378 IC50 = 22000 nM T20251 CA72PE 49847379 IC50 = 46000 nM T20251 C4V7EW 49848258 IC50 = 19000 nM T20251 C4BXP1 49848557 IC50 > 50118.72 nM T20251 CP8TS6 49848895 IC50 = 6400 nM T20251 C9COF5 49848896 IC50 = 23000 nM T20251 CK0B1G 49848897 IC50 = 13000 nM T20251 CP61VJ 49849002 IC50 = 31000 nM T20251 CBM62Z 49849007 IC50 = 54000 nM T20251 C05SEW 49849008 IC50 = 7200 nM T20251 CF64IJ 49849120 IC50 = 38000 nM T20251 CC9EB4 49849122 IC50 = 21000 nM T20251 C2ORV5 49849123 IC50 = 2000 nM T20251 CTR7Q0 49850345 IC50 > 50118.72 nM T20251 CSGQ38 49850568 Ki = 316.23 nM T20251 C07JTU 49850570 Ki = 630.96 nM T20251 CR4EZ0 49850870 Ki = 501.19 nM T20251 C5K4EC 49850872 Ki = 3981.07 nM T20251 C8AW0R 49850874 Ki = 50.12 nM T20251 CL59YO 49852191 IC50 > 30000 nM T20251 C7ZUF5 49852192 IC50 > 30000 nM T20251 C6KX1V 49852195 IC50 > 30000 nM T20251 CN2V8R 49854681 IC50 = 5700 nM T20251 C65YMH 49855492 IC50 > 33000 nM T20251 C12FKR 49855495 IC50 = 19000 nM T20251 CP3M8H 49855496 IC50 > 33000 nM T20251 CKT38C 49855683 IC50 > 33000 nM T20251 C8KA3J 49855886 IC50 > 33000 nM T20251 C9TO2S 49856484 IC50 = 4800 nM T20251 C6UO5Y 49857245 IC50 = 1500 nM T20251 C0UOW3 49857439 IC50 = 11100 nM T20251 CQ3LC1 49857440 IC50 = 2300 nM T20251 CW9NX3 49858377 IC50 > 33000 nM T20251 C1EMQ2 49861348 Ki > 10 nM T20251 CR53VH 49862169 Ki = 2160 nM T20251 CT3WH4 49862215 Ki = 1580 nM T20251 CC97JM 49862219 Ki = 1780 nM T20251 C6IW4Q 49862238 Ki > 1000 nM T20251 CB13XF 49863795 IC50 = 700 nM T20251 C18ICN 49863958 IC50 = 11800 nM T20251 CMRQ30 49863961 IC50 = 6900 nM T20251 CLOY62 49864459 IC50 > 10000 nM T20251 CR8JK9 49864483 IC50 > 10000 nM T20251 C0Y5ZU 49865137 IC50 > 10000 nM T20251 CG98LM 49865191 IC50 > 10000 nM T20251 CKWA93 49865589 IC50 > 63095.73 nM T20251 CXWL20 49865623 IC50 = 1584.89 nM T20251 CXW97O 49865703 IC50 > 33000 nM T20251 CRG60N 49865732 IC50 > 33000 nM T20251 CZY2T3 49865733 IC50 = 0.61 nM T20251 CI2W0D 49865783 IC50 = 250 nM T20251 CUK35O 49865784 IC50 = 1100 nM T20251 CLD4P0 49865785 IC50 = 20000 nM T20251 CFZ39O 49865822 IC50 = 3100 nM T20251 CL0DR3 49865859 IC50 = 1100 nM T20251 CE15WQ 49865860 IC50 = 1000 nM T20251 C4EM1X 49865861 IC50 = 1600 nM T20251 CEF3O1 49865862 IC50 = 1500 nM T20251 C5YP2L 49865863 IC50 = 1000 nM T20251 CK7O1S 49865875 IC50 > 10000 nM T20251 C8V3NG 49865877 IC50 > 10000 nM T20251 CEK89Q 49865878 IC50 > 10000 nM T20251 CZA5X4 49865879 IC50 > 10000 nM T20251 CD4LO5 49865880 IC50 > 10000 nM T20251 CNGL32 49865918 IC50 = 15000 nM T20251 C9HEP1 49865919 IC50 = 680 nM T20251 CL6ZG8 49865920 IC50 = 660 nM T20251 CHYN61 49865922 IC50 = 1100 nM T20251 C3YJ4G 49865936 IC50 > 10000 nM T20251 CB5WR8 49865937 IC50 = 5900 nM T20251 C5NJ6K 49865969 IC50 = 340 nM T20251 C3CJ4R 49865970 IC50 = 680 nM T20251 CP8VQ6 49865971 IC50 = 1000 nM T20251 CAI09G 49865972 IC50 = 1400 nM T20251 C5TMG9 49865973 IC50 = 1300 nM T20251 CFT26X 49866025 IC50 = 1600 nM T20251 CN9PI1 49867423 Ki = 120 nM T20251 CMV6Y2 49868651 IC50 = 4100 nM T20251 C8AJ5K 49869035 IC50 = 16700 nM T20251 C1WM9N 49869037 IC50 > 33000 nM T20251 CAPI06 49869040 IC50 = 28800 nM T20251 CG5IV6 49869041 IC50 = 21000 nM T20251 C1WYF9 49869172 IC50 > 33000 nM T20251 CR0D3P 49869174 IC50 > 33000 nM T20251 C19EDA 49869312 IC50 = 12400 nM T20251 CD62TH 49869313 IC50 = 14400 nM T20251 CMB32F 49869877 IC50 = 24500 nM T20251 C07DIE 49870853 IC50 > 63000 nM T20251 C7GR0H 49872381 IC50 = 7900 nM T20251 CD1X3U 49872384 IC50 > 10000 nM T20251 C60RMP 49872483 IC50 > 10000 nM T20251 CD5J7W 50898619 IC50 = 4100 nM T20251 CX5V7B 50898694 IC50 = 15400 nM T20251 C90UKY 50899643 IC50 = 16000 nM T20251 CYGD56 50899654 IC50 > 10000 nM T20251 CBLK68 50899745 IC50 = 5400 nM T20251 CU7TK4 50899749 IC50 > 10000 nM T20251 C1R5UC 50905013 Ki = 27000 nM T20251 C67IRJ 50908804 Ki = 2511.89 nM T20251 CLOB24 50908805 Ki = 1995.26 nM T20251 CL01TJ 50913783 IC50 = 3800 nM T20251 C1YF6I 50915132 IC50 > 30000 nM T20251 CD0G9L 50915507 IC50 = 10000 nM T20251 C4IOV5 50916528 IC50 > 30000 nM T20251 C7JB8Z 50925394 IC50 < 1000 nM T20251 CP2N7E 50925496 Ki = 14000 nM T20251 CX3NI6 50925497 Ki = 16000 nM T20251 C64HTN 50925513 IC50 = 3500 nM T20251 C2GTE4 50938548 IC50 = 1600 nM T20251 C90ANW 50939489 IC50 = 6900 nM T20251 CJ43IF 50941460 IC50 = 7800 nM T20251 C2HJL6 50942025 IC50 = 2230 nM T20251 CP7B9V 50942696 IC50 = 3900 nM T20251 COJ32C 50942806 IC50 >= 10000 nM T20251 CWK9X2 50942874 IC50 >= 10000 nM T20251 CX8N4D 50990920 IC50 = 8000 nM T20251 CXF4V3 50990921 IC50 = 65000 nM T20251 C2T4IC 50991056 IC50 = 31300 nM T20251 CI32TR 50992246 IC50 = 1700 nM T20251 C4IFR9 50992499 IC50 = 2000 nM T20251 CFG8M7 50992643 IC50 = 10 nM T20251 C41QJN 50992719 IC50 = 1000 nM T20251 C4BP6M 50992720 IC50 = 5000 nM T20251 CIO9B5 50992721 IC50 = 6000 nM T20251 C2ST3V 50992722 IC50 = 5000 nM T20251 C2SHO8 50993865 IC50 = 1600 nM T20251 CLY9W1 50994950 IC50 = 8300 nM T20251 C2CH1R 50995330 IC50 > 30000 nM T20251 C0X9OY 50997095 IC50 = 49 nM T20251 CS9G6E 50997096 IC50 = 460 nM T20251 C4UPJ2 51030637 IC50 = 10000 nM T20251 CP6NI2 51030711 IC50 > 9800 nM T20251 CSE2G4 51030732 IC50 = 500 nM T20251 CM1F2R 51030830 IC50 = 1900 nM T20251 CWQ20B 51030833 IC50 = 2000 nM T20251 C15LDS 51030834 IC50 = 800 nM T20251 C1P9UY 51030897 IC50 = 5900 nM T20251 CW06HL 51030898 IC50 = 11600 nM T20251 C4QW2B 51030901 IC50 = 7600 nM T20251 C48USP 51030919 IC50 = 1900 nM T20251 C0QP3A 51030920 IC50 = 80000 nM T20251 C70OGS 51030984 IC50 = 12000 nM T20251 CX28ZP 51030985 IC50 = 10000 nM T20251 CXB2Q6 51031001 IC50 > 30000 nM T20251 CUY1S2 51033690 IC50 = 17000 nM T20251 CVE0J3 51033997 IC50 > 20000 nM T20251 CAU5Y8 51038251 IC50 = 1820 nM T20251 CBA1X5 51039205 IC50 = 32100 nM T20251 C96AQN 51346908 IC50 = 28900 nM T20251 C2W8LE 51346934 IC50 > 10000 nM T20251 CA3Y7Q 51347395 IC50 = 0.66 ug.mL-1 T20251 C3MWD8 51349244 IC50 = 2630 nM T20251 CO7U5C 51355838 IC50 = 15000 nM T20251 CIXL91 51355841 IC50 > 30000 nM T20251 C3XQE2 52337837 IC50 = 5 nM T20251 C8K6CQ 52916803 IC50 = 68000 nM T20251 CIRP71 52917998 IC50 = 2 nM T20251 CT0B1S 52917999 IC50 = 290 nM T20251 CFX76G 52918016 IC50 = 140 nM T20251 C47RHB 52918017 IC50 = 1260 nM T20251 CUQ53T 52918018 IC50 = 10000 nM T20251 CTP6U5 52918019 IC50 > 10000 nM T20251 CTJ28K 52918135 IC50 > 20000 nM T20251 CCP0V7 52920236 IC50 = 4000 nM T20251 CKDE49 52933949 IC50 = 21000 nM T20251 CL2Q9F 52934178 IC50 = 23000 nM T20251 CDI09M 52934690 IC50 = 5100 nM T20251 CUV9B4 52934924 IC50 = 12900 nM T20251 CEMS67 52938764 IC50 > 100000 nM T20251 CJ19FP 52940753 IC50 = 199.53 nM T20251 CCDZ51 52940788 IC50 = 1258.93 nM T20251 CH5S0P 52940936 Ki > 10000 nM T20251 C2RW5A 52940961 IC50 = 5011.87 nM T20251 CKP92N 52941058 Ki = 500 nM T20251 C8FZL4 52941427 IC50 = 794.33 nM T20251 COK7Q1 52941460 Ki > 20000 nM T20251 C1M3SD 52941462 IC50 = 0.38 nM T20251 CUV8I6 52941526 IC50 = 12100 nM T20251 C58ART 52941549 IC50 = 15 nM T20251 CVT1A7 52941563 Ki = 11000 nM T20251 C7N6RA 52941564 Ki > 20000 nM T20251 CP8BI3 52941601 IC50 = 1200 nM T20251 C1FX6A 52941684 IC50 > 63000 nM T20251 CE26GV 52941856 IC50 = 5900 nM T20251 C5JAY6 52941880 IC50 > 10000 nM T20251 CU7A2Y 52941972 IC50 = 1000 nM T20251 C51MIQ 52942095 Ki = 710 nM T20251 C0OU8I 52942126 IC50 = 740 nM T20251 C3E5WI 52942171 Ki = 2510 nM T20251 CL65FB 52942200 Ki = 560 nM T20251 C3WH6F 52942248 Ki = 1120 nM T20251 CYLC29 52942529 IC50 = 4.6 nM T20251 CX9AF4 52942551 Ki = 3162.28 nM T20251 CPOQ82 52942580 IC50 = 1.9 nM T20251 C3YF5D 52942581 IC50 = 7.3 nM T20251 CR0G5U 52942644 Ki > 31622.78 nM T20251 CKN2U6 52942810 IC50 = 3.7 nM T20251 CX2E5H 52942854 Ki = 969 nM T20251 C8N4AB 52943069 IC50 > 10000 nM T20251 C5V4DW 52943162 IC50 = 0.14 nM T20251 C2DOU4 52943195 IC50 = 400 nM T20251 CXD0O1 52943196 IC50 = 20000 nM T20251 CNI79L 52943227 Ki = 370 nM T20251 C0F3LG 52943305 IC50 = 3200 nM T20251 CJWI80 52943409 Ki > 10000 nM T20251 C71MDG 52943756 IC50 < 1000 nM T20251 CNK14O 52943803 IC50 = 0.62 nM T20251 CCF97B 52943811 Ki = 25118.86 nM T20251 C2FG9O 52943861 Ki = 31622.78 nM T20251 C9G4CI 52943891 Ki = 7943.28 nM T20251 CRH1Q5 52943993 IC50 = 4.8 nM T20251 CBW0A9 52944041 IC50 = 1.8 nM T20251 CE7K2D 52944154 IC50 = 260 nM T20251 C25NCO 52944522 Ki = 3980 nM T20251 C89GIK 52944552 IC50 = 3.5 nM T20251 CO85FM 52944637 Ki = 400 nM T20251 CCVP06 52944840 Ki = 5011.87 nM T20251 CP5A3T 52944907 IC50 = 13 nM T20251 C54ZBG 52944974 IC50 = 3 nM T20251 CQJ7C0 52945023 IC50 = 1000 nM T20251 CV48KS 52945118 IC50 = 0.72 nM T20251 C1G0IP 52945138 IC50 = 6 nM T20251 C34ZMB 52945520 IC50 > 30000 nM T20251 CSZ4R3 52945588 IC50 = 0.25 nM T20251 CNGU78 52945626 IC50 = 0.52 nM T20251 C1Z9HY 52945786 Ki > 10000 nM T20251 C5RAX8 52945794 IC50 > 100000 nM T20251 CF46DK 52945849 Ki = 320 nM T20251 CNQF49 52945978 IC50 = 63095.73 nM T20251 CJ49MX 52946290 Ki = 5011.87 nM T20251 CG8CN4 52946340 IC50 > 33 nM T20251 CK5VU2 52946383 IC50 > 63000 nM T20251 COZ9J3 52946432 IC50 = 2511.89 nM T20251 C4K6BH 52946883 Ki > 10000 nM T20251 C2GVW6 52947078 Ki > 10000 nM T20251 CK5ER0 52947414 Ki = 3981.07 nM T20251 CFD18K 52947437 IC50 > 33 nM T20251 CI5V3X 52947507 IC50 = 5011.87 nM T20251 CFN7I8 52947509 IC50 = 3.3 nM T20251 C6ZSQ8 52947516 IC50 = 1995.26 nM T20251 C41AYU 52947523 IC50 > 33 nM T20251 CEU2N1 52947551 IC50 = 12600 nM T20251 CY06OH 52947573 IC50 = 1.6 nM T20251 CY72CQ 52947593 IC50 = 4.9 nM T20251 CAVB03 52947615 Ki = 10000 nM T20251 CCIG41 52947616 IC50 = 1400 nM T20251 CGCK63 52947618 IC50 > 63000 nM T20251 C1HRK4 52947622 Ki = 6309.57 nM T20251 CN32PV 52947694 IC50 = 1584.89 nM T20251 CFI96N 52947735 IC50 = 0.62 nM T20251 CI63UL 52948240 IC50 = 1.5 nM T20251 CZ01DH 52948653 IC50 = 6309.57 nM T20251 C15KNW 52948655 IC50 = 13 nM T20251 C4ZC1K 52948697 Ki = 3981.07 nM T20251 C48RBH 52948719 IC50 = 0.43 nM T20251 CZX5B9 52948735 IC50 = 6.6 nM T20251 CDN06O 52948827 IC50 > 63000 nM T20251 CE0R3S 52948850 IC50 = 4.7 nM T20251 C25FAX 52948924 Ki = 3160 nM T20251 CPN4Z8 52948969 IC50 = 2.8 nM T20251 CN85WP 52949210 IC50 = 4800 nM T20251 CH02CI 52949290 IC50 = 800 nM T20251 C9OSI0 52949300 IC50 = 630.96 nM T20251 C9YWD1 52949393 Ki > 10000 nM T20251 CROV43 52949411 Ki > 10000 nM T20251 C0AZH4 52949420 Ki = 630 nM T20251 CVWY23 52949439 IC50 = 2.8 nM T20251 CRL18H 52949508 Ki = 1580 nM T20251 C9V6GB 52950007 IC50 = 0.95 nM T20251 C4OAP3 53234015 IC50 > 5000 nM T20251 CT3F0N 53235532 Ki = 700 nM T20251 C8ETM0 53237536 IC50 = 390 nM T20251 CYHS15 53237773 IC50 = 2000 nM T20251 C8EW1X 53239080 IC50 < 30000 nM T20251 CFI32H 53239287 Ki = 11600 nM T20251 CMYJ58 53239519 IC50 < 30000 nM T20251 CMQZ70 53242178 IC50 > 100000 nM T20251 CKNJ47 53245660 IC50 > 33000 nM T20251 CW9IQ0 53248730 IC50 > 33000 nM T20251 CQIY23 53248846 IC50 > 60000 nM T20251 C9MHR0 53248847 IC50 = 25000 nM T20251 CG3LA9 53248849 IC50 = 1890 nM T20251 CNB90W 53257735 IC50 = 19054.61 nM T20251 CW0M1K 53259021 IC50 = 1000 nM T20251 C70QNI 53260398 IC50 = 1000 nM T20251 C9NF0C 53302364 IC50 > 30000 nM T20251 CRB6N5 53307604 IC50 > 26302.68 nM T20251 CWQ8Y2 53307787 IC50 = 390 nM T20251 CR7TD8 53307788 IC50 > 10000 nM T20251 CQ87XN 53307874 Ki = 800 nM T20251 CW4S5E 53307875 Ki = 250 nM T20251 C7V1YI 53307876 Ki = 1100 nM T20251 C6QY4D 53307877 Ki = 1900 nM T20251 C68TEC 53307957 Ki = 970 nM T20251 CY92LZ 53310757 IC50 > 10000 nM T20251 CDT9H2 53310826 IC50 = 4300 nM T20251 CLZ60N 53310827 IC50 > 30000 nM T20251 C06JVE 53310828 IC50 > 30000 nM T20251 CZ6T1A 53310829 IC50 = 7100 nM T20251 CE9UD4 53310977 IC50 > 30000 nM T20251 C1O8DZ 53310978 IC50 > 30000 nM T20251 CCV51N 53310979 IC50 > 30000 nM T20251 C38JFV 53310980 IC50 > 30000 nM T20251 CR97IC 53310981 IC50 > 30000 nM T20251 CI6J2A 53310982 IC50 > 30000 nM T20251 C19ZEA 53311068 IC50 = 20500 nM T20251 CQ7B4Z 53311133 IC50 = 3000 nM T20251 CRI92N 53311230 IC50 > 50118.72 nM T20251 CJ83EB 53311393 IC50 = 4700 nM T20251 CG5WV2 53312065 IC50 = 9700 nM T20251 C89ETA 53312066 IC50 > 11000 nM T20251 CZ5IB8 53312148 IC50 > 11000 nM T20251 CVW9A8 53312150 IC50 > 11000 nM T20251 C9P4YV 53316457 IC50 = 3830 nM T20251 CW7TF1 53316459 IC50 = 1160 nM T20251 C1-MAY-02 53317017 IC50 > 10000 nM T20251 CPS12B 53317097 IC50 > 10000 nM T20251 CHNX58 53317305 IC50 = 4.3 nM T20251 CDH87Y 53317306 IC50 = 2.9 nM T20251 CK3MZ0 53317307 IC50 = 0.67 nM T20251 C9RK8W 53317504 IC50 = 1120 nM T20251 CNZ84M 53317555 IC50 = 6025.6 nM T20251 CK27PC 53317643 IC50 = 7300 nM T20251 CXV3W2 53317718 Ki > 60000 nM T20251 CP14EK 53317957 Ki = 35000 nM T20251 CL45CT 53318503 IC50 = 4300 nM T20251 C13SNK 53318592 IC50 > 10 nM T20251 CGWD27 53318593 IC50 = 2.4 nM T20251 C54SRN 53318594 IC50 = 7 nM T20251 C74CVF 53318595 IC50 = 1.7 nM T20251 C37ZAQ 53318697 IC50 = 4730 nM T20251 CBLD50 53318698 IC50 = 390 nM T20251 CK1ZI3 53318801 IC50 > 10 nM T20251 CB09MA 53318910 IC50 = 21000 nM T20251 CK2G3D 53319480 IC50 = 2000 nM T20251 CTA23R 53319654 IC50 = 7800 nM T20251 CUG7V3 53320013 IC50 = 990 nM T20251 CS04NZ 53320014 IC50 = 300 nM T20251 CTJ59M 53320020 Ki = 1621 nM T20251 CWLQ84 53320117 IC50 = 9.3 nM T20251 CVU69D 53320143 IC50 = 251.19 nM T20251 CGZX46 53320144 IC50 = 17.78 nM T20251 CXF1S4 53320328 IC50 = 1610 nM T20251 CB84NG 53320778 IC50 = 2320 nM T20251 CML70D 53321223 IC50 = 0.81 nM T20251 CQD62W 53321323 IC50 = 980 nM T20251 COT69M 53321324 IC50 = 510 nM T20251 CAJ4L7 53321331 Ki = 119 nM T20251 CJ9BK7 53321473 IC50 = 83176.38 nM T20251 C7Y2AB 53321474 IC50 = 74131.02 nM T20251 CRY96M 53321650 Ki = 3162.28 nM T20251 C4X3IS 53321979 IC50 = 3500 nM T20251 CMH54U 53322279 IC50 = 7600 nM T20251 C3YWZ5 53322451 IC50 = 40000 nM T20251 C98PDX 53322555 IC50 = 1.9 nM T20251 C5G8RQ 53322642 Ki = 7080 nM T20251 C1WA2E 53322643 Ki = 3802 nM T20251 C35XLW 53322810 IC50 = 4900 nM T20251 C01ILC 53322949 IC50 = 3162.28 nM T20251 CGN6Z3 53323531 Ki = 1.3 nM T20251 CR57HN 53323639 IC50 = 1400 nM T20251 CX54CT 53323813 IC50 = 23000 nM T20251 CDRV76 53323814 IC50 = 23000 nM T20251 C8ZHY7 53323979 IC50 = 310 nM T20251 C0HC8D 53324076 IC50 = 1.2 nM T20251 C1VNZ9 53324198 IC50 = 5000 nM T20251 CC08MY 53324265 IC50 > 20000 nM T20251 C2XT7J 53324382 IC50 = 107.15 nM T20251 C4ZO1H 53324408 IC50 = 2270 nM T20251 CS3L5G 53325164 IC50 = 4.3 nM T20251 CUO1R8 53325274 IC50 > 10000 nM T20251 CZB7M2 53325275 IC50 = 140 nM T20251 C3QNR2 53325463 IC50 = 3250 nM T20251 CZN8B4 53325581 IC50 = 5270 nM T20251 COS87G 53325596 IC50 = 102329.3 nM T20251 CY15EU 53325639 IC50 = 3900 nM T20251 CZ1SE0 53325908 Ki > 60000 nM T20251 C1N7XO 53325966 IC50 = 8600 nM T20251 CYA3F1 53325983 IC50 = 1500 nM T20251 C28HNA 53326213 IC50 > 10000 nM T20251 C9ZF4V 53326457 IC50 = 5.8 nM T20251 C3KWC5 53326627 IC50 > 10000 nM T20251 C5O1VT 53326682 IC50 = 537031.8 nM T20251 C0K7AS 53326693 IC50 = 218776.16 nM T20251 C18TPG 53326909 IC50 = 40000 nM T20251 C1KYR9 53326941 IC50 = 2600 nM T20251 CUF26V 53326945 IC50 = 501.19 nM T20251 C7J8ZY 53327611 IC50 = 13600 nM T20251 CQ7LB1 53327841 IC50 > 30000 nM T20251 CC6ME0 53327888 IC50 > 30000 nM T20251 C9F7ED 53341130 Ki = 1254 nM T20251 CCX7M5 53353847 IC50 > 30000 nM T20251 CS4HK7 53354783 IC50 = 170 nM T20251 C8PJ6E 53354789 IC50 = 40000 nM T20251 CYMP74 53354793 IC50 = 20000 nM T20251 C8ZRE3 53356518 IC50 > 80000 nM T20251 C6O7VL 53357600 IC50 = 25900 nM T20251 CYG6Q1 53358318 IC50 = 2600 nM T20251 C3B5AJ 53361011 IC50 > 30000 nM T20251 C9H5YE 53361128 IC50 > 10000 nM T20251 C23WVS 53361524 IC50 > 10000 nM T20251 CX83CK 53362097 IC50 = 5600 nM T20251 C54YUZ 53362500 IC50 > 10000 nM T20251 C6CR4I 53362501 IC50 = 1930 nM T20251 CJW0B3 53362502 IC50 = 440 nM T20251 CBAC86 53362558 IC50 = 4100 nM T20251 CYX87Q 53362559 IC50 = 2600 nM T20251 C8B1ZY 53362973 IC50 = 3800 nM T20251 COG5K0 53363092 IC50 = 7520 nM T20251 CCZW39 53363093 IC50 = 8160 nM T20251 CU59EZ 53363442 IC50 = 10000 nM T20251 C1PVA2 53363480 Ki = 6309.57 nM T20251 CU7VZ1 53363805 IC50 = 5770 nM T20251 C4D9RH 53363970 IC50 = 8480 nM T20251 C6N8KX 53363971 IC50 = 31240 nM T20251 C3WBV5 53364352 IC50 > 30000 nM T20251 CSV85J 53364356 IC50 = 10400 nM T20251 C2PHM7 53364357 IC50 = 10030 nM T20251 CNI7P9 53372541 IC50 = 10000 nM T20251 CA6H2P 53372668 IC50 = 398.11 nM T20251 CFM7W8 53372672 IC50 = 31622.78 nM T20251 C9GYZ3 53372790 IC50 = 3162.28 nM T20251 CT6K2O 53373472 IC50 = 15000 nM T20251 CL37YO 53380288 IC50 > 10000 nM T20251 C4ORN7 53380491 IC50 > 30000 nM T20251 CK52GI 53380818 IC50 > 30000 nM T20251 CZWO31 53387025 EC50 = 4700 nM T20251 C87NKH 53387026 IC50 = 4700 nM T20251 CCUH12 53387402 IC50 > 30000 nM T20251 CJ39QE 53387563 IC50 = 5700 nM T20251 CI15GW 53387564 IC50 = 21000 nM T20251 CS7X9W 53387565 IC50 = 5600 nM T20251 CIGM78 53389570 IC50 > 30000 nM T20251 CVG90B 53389651 IC50 > 10000 nM T20251 C47VGW 53393916 IC50 > 20000 nM T20251 C1QYU2 53464257 Ki = 5600 nM T20251 C6KC5V 53464567 Ki > 15000 nM T20251 C4Q0JV 53464571 Ki > 15000 nM T20251 CPE0Q3 53464695 Ki > 10000 nM T20251 CG7NH3 53464819 Ki = 2770 nM T20251 CC7P2U 53464882 Ki > 15000 nM T20251 CPRZ03 53464941 Ki > 10000 nM T20251 CRA3L0 53464942 Ki > 15000 nM T20251 CYE6O4 53464943 Ki > 10000 nM T20251 C3I8KD 53464944 Ki > 15000 nM T20251 C6K5JY 53464945 Ki > 10000 nM T20251 CK8YI4 53465003 Ki > 15000 nM T20251 C9K6FT 53465005 Ki > 15000 nM T20251 CH9CX8 53465067 Ki > 10000 nM T20251 CVM91G 53465142 Ki > 15000 nM T20251 C24FQU 53465297 IC50 = 9100 nM T20251 CHN72W 53469852 IC50 = 4200 nM T20251 CK1C9O 53472113 IC50 = 1400 nM T20251 CH5A9S 53484202 IC50 = 12080 nM T20251 CG3FA9 53492750 IC50 = 12882.5 nM T20251 C4U5IX 53493001 EC50 = 15000 nM T20251 CE9K7U 53494972 IC50 = 53000 nM T20251 C7TR2W 53497131 IC50 = 25100 nM T20251 CWA14L 53802926 IC50 = 6309.57 nM T20251 CP24ZC 54579002 IC50 = 8700 nM T20251 CTA9K1 54579972 IC50 = 45 nM T20251 C1GXF9 54579973 IC50 = 370 nM T20251 CQ8AZ0 54580065 Ki = 1584.89 nM T20251 CYM8N2 54580066 Ki = 794.33 nM T20251 CT2FB8 54580068 Ki = 1995.26 nM T20251 C4KGT2 54580069 Ki = 2511.89 nM T20251 CL5V4H 54580071 Ki = 316.23 nM T20251 CG86QM 54580083 IC50 = 56234.13 nM T20251 C4RH7W 54580091 IC50 = 18197.01 nM T20251 CC0R4A 54580092 IC50 > 31622.78 nM T20251 C73HNQ 54580097 IC50 = 41686.94 nM T20251 C89MEB 54580190 IC50 = 8600 nM T20251 CMDO43 54580283 Ki = 80 nM T20251 C6M4ND 54580284 Ki = 40 nM T20251 CB58LO 54580324 IC50 = 8912.51 nM T20251 CLW26Q 54580457 IC50 = 160 nM T20251 CRV6M8 54580555 IC50 = 900 nM T20251 C2YWA6 54580845 IC50 = 8620 nM T20251 C6R3MZ 54580973 IC50 = 790 nM T20251 C4GAB9 54581050 Ki = 1584.89 nM T20251 CP7HC3 54581052 Ki = 2511.89 nM T20251 CF9L7B 54581072 IC50 = 44668.36 nM T20251 C54SOM 54581080 IC50 > 50118.72 nM T20251 CC3J5L 54581190 IC50 = 7600 nM T20251 C8S1LG 54581286 Ki = 80 nM T20251 CQ6V1E 54581466 IC50 = 1030 nM T20251 C4EH1F 54581551 IC50 = 440 nM T20251 CBT56Y 54581676 IC50 = 2300 nM T20251 CJV9G1 54581702 IC50 = 3200 nM T20251 CQ0YA3 54581861 IC50 = 1890 nM T20251 CHJK47 54581904 IC50 = 6230 nM T20251 C7QWE4 54581905 IC50 = 9400 nM T20251 C8CTD7 54581962 IC50 = 1200 nM T20251 CUN59X 54582014 IC50 = 28 nM T20251 C5S1ZK 54582015 IC50 = 1960 nM T20251 CWKA42 54582019 IC50 = 2000 nM T20251 CL52TN 54582094 Ki = 251.19 nM T20251 CB6DW8 54582096 Ki = 630.96 nM T20251 C10TMQ 54582108 IC50 = 31622.78 nM T20251 C69IDP 54582109 IC50 = 1995.26 nM T20251 C5Y1OZ 54582114 IC50 > 50118.72 nM T20251 CG3HB9 54582215 IC50 = 2100 nM T20251 C4KMX1 54582216 IC50 = 8900 nM T20251 CD1AE2 54582217 IC50 = 6500 nM T20251 CAG68L 54582303 Ki = 200 nM T20251 C51QIK 54582357 IC50 = 7943.28 nM T20251 C1HBD8 54582798 IC50 = 16000 nM T20251 CB8JV7 54582823 IC50 = 7110 nM T20251 CZ71VB 54582892 IC50 > 30000 nM T20251 C2CAO0 54582957 IC50 = 200 nM T20251 CZ3DW2 54582958 IC50 = 47 nM T20251 CS3P4K 54582960 IC50 = 29 nM T20251 CD0WT4 54582961 IC50 = 16 nM T20251 CP8TG1 54583028 Ki = 251.19 nM T20251 CHT78R 54583030 Ki = 630.96 nM T20251 CUHW91 54583050 IC50 = 1584.89 nM T20251 CX24KS 54583051 IC50 = 50118.72 nM T20251 CB8S6F 54583055 IC50 > 31622.78 nM T20251 C14MKQ 54583056 IC50 = 794.33 nM T20251 CUC32E 54583059 IC50 = 52480.75 nM T20251 CLX7U9 54583111 IC50 = 17000 nM T20251 C3WZ9I 54583112 IC50 = 52800 nM T20251 CYD20W 54583185 IC50 = 42600 nM T20251 COQD25 54583186 IC50 = 1200 nM T20251 CC19ZA 54583187 IC50 = 300 nM T20251 CEOZ15 54583522 IC50 = 12500 nM T20251 CXLA39 54583624 IC50 = 30000 nM T20251 C9OB1C 54583833 IC50 = 6670 nM T20251 CE61RX 54583834 IC50 = 5200 nM T20251 CG78OW 54583895 IC50 = 5400 nM T20251 CSCE48 54583896 IC50 = 1500 nM T20251 C6UED1 54583954 IC50 = 56 nM T20251 CU10AQ 54584056 IC50 = 79432.82 nM T20251 CUKW62 54584057 IC50 = 63095.73 nM T20251 CDV2Z9 54584068 IC50 = 30902.95 nM T20251 C90AHI 54584164 IC50 = 3900000 nM T20251 C7MP0S 54584254 Ki = 4168.69 nM T20251 CY80OU 54584273 Ki = 500 nM T20251 C8YEA3 54584294 IC50 = 30199.52 nM T20251 C4LN8M 54584295 IC50 = 12882.5 nM T20251 CVUI69 54584296 IC50 = 100000 nM T20251 CJV94T 54584501 IC50 = 3400 nM T20251 CPS93U 54584537 IC50 < 200 nM T20251 CTM3D4 54584797 IC50 = 3850 nM T20251 CF49IN 54584798 IC50 = 18800 nM T20251 C3C8QF 54584905 IC50 = 34 nM T20251 C7UY2T 54584908 IC50 = 28 nM T20251 CR7UW2 54584957 IC50 = 31622.78 nM T20251 C8P6MI 54584991 Ki = 1000 nM T20251 CI0P4H 54585005 IC50 = 125892.54 nM T20251 CZ4S0B 54585107 IC50 > 90000 nM T20251 C3TAR4 54585108 IC50 = 35900 nM T20251 C8RTU2 54585109 IC50 < 300 nM T20251 CL7P1G 54585233 Ki = 5011.87 nM T20251 C9PB7S 54585251 IC50 = 36307.81 nM T20251 C30LYP 54585371 Ki = 630.96 nM T20251 C2A6ER 54585480 IC50 < 200 nM T20251 CY5LT9 54585737 IC50 = 18600 nM T20251 C0C2BE 54585833 IC50 = 600 nM T20251 CPX76L 54585862 IC50 = 20300 nM T20251 CW31VH 54585863 IC50 = 120 nM T20251 C2M9RO 54585864 IC50 = 4620 nM T20251 C8OR2E 54585941 Ki = 3981.07 nM T20251 C4V8AE 54585969 IC50 = 25118.86 nM T20251 CN8E3L 54585970 IC50 = 6025.6 nM T20251 CJ4QK6 54585971 IC50 = 63095.73 nM T20251 CH6X1P 54585974 IC50 > 31622.78 nM T20251 CC6HY7 54586021 IC50 = 1100 nM T20251 C3MLH7 54586172 Ki = 1584.89 nM T20251 CSX84E 54586210 IC50 = 10000 nM T20251 CSC0H3 54586414 IC50 = 16400 nM T20251 C7HD0U 54586415 IC50 = 1500 nM T20251 C8TLD6 54586719 IC50 = 2150 nM T20251 CYVZ19 54586720 IC50 = 2180 nM T20251 C67NFK 54586780 IC50 = 10600 nM T20251 C4ACJ8 54586781 IC50 = 4000 nM T20251 C59FXV 54586919 Ki = 1258.93 nM T20251 CTK5S1 54586921 Ki = 794.33 nM T20251 CCL0M3 54586940 IC50 = 25118.86 nM T20251 C6VQT3 54587171 Ki = 150 nM T20251 CSX1R5 54587172 Ki = 3700 nM T20251 CO19MR 54587173 Ki = 2300 nM T20251 CLAJ60 54587208 Ki = 1258.93 nM T20251 C09OSL 54587230 IC50 = 12022.64 nM T20251 C0UYD7 54587231 IC50 = 8912.51 nM T20251 CD06RB 54587434 IC50 = 24400 nM T20251 C8MH6B 54587759 IC50 = 27000 nM T20251 CH3US7 54587760 IC50 > 33000 nM T20251 CZ5IY9 54587813 IC50 = 2600 nM T20251 C30XLO 54592009 IC50 > 100000 nM T20251 C57DQW 54670057 IC50 = 100 nM T20251 C7L5YB 54670058 IC50 = 39 nM T20251 CM7FC6 54670152 IC50 = 780 nM T20251 CF7XA0 54674257 IC50 = 21000 nM T20251 C3S9EC 54674292 IC50 = 12140 nM T20251 C9JCZ5 54675567 IC50 = 2780 nM T20251 C0ZG2V 54709839 IC50 = 20000 nM T20251 CO75TL 54712015 IC50 > 50000 nM T20251 CLT3Q8 54716246 IC50 > 10000 nM T20251 C28RDF 54746913 IC50 > 60000 nM T20251 C5OBC3 54753437 IC50 > 10000 nM T20251 CGIP16 54754722 IC50 = 32000 nM T20251 CX4LK5 54754723 IC50 = 5600 nM T20251 C6LZ8B 54754724 IC50 = 5000 nM T20251 CSA9I6 54754844 IC50 = 24000 nM T20251 CEGJ53 54754845 IC50 = 32000 nM T20251 C9NV8L 54754967 IC50 = 32000 nM T20251 CI78YZ 54754968 IC50 = 2500 nM T20251 CV3K8U 54754969 IC50 = 1100 nM T20251 C6T8XS 54755079 IC50 = 9500 nM T20251 CL2AU5 54755081 IC50 = 9100 nM T20251 C2R6KO 54755083 IC50 = 34000 nM T20251 C5LT0A 54755193 IC50 = 6200 nM T20251 C3SD6W 54755560 IC50 = 7600 nM T20251 C4GBT5 54755562 IC50 = 2500 nM T20251 C0KZ4M 54755801 IC50 = 7600 nM T20251 C2QP4W 54755919 IC50 = 1900 nM T20251 CPWZ05 54756038 IC50 = 5600 nM T20251 CJBW64 54756045 IC50 = 20000 nM T20251 C0ZWL2 54756156 IC50 = 3700 nM T20251 CI20JA 54756906 IC50 = 6760.83 nM T20251 CCG08B 54756907 IC50 = 12589.25 nM T20251 CK50BF 54756908 IC50 = 19952.62 nM T20251 CILG27 54758399 IC50 = 17782.79 nM T20251 C8AB1J 54759606 IC50 = 18830 nM T20251 C80STN 54761221 IC50 > 10000 nM T20251 C0Y9ZG 54761473 IC50 = 15000 nM T20251 CU62DN 54764919 IC50 > 10000 nM T20251 C0T3KY 54765285 IC50 = 3700 nM T20251 CFHI34 54768835 IC50 = 8300 nM T20251 CLY35F 54768836 IC50 = 2100 nM T20251 C9U4YQ 54768838 IC50 = 25700 nM T20251 CO4FY1 54769305 IC50 = 5200 nM T20251 CFC91M 54769914 IC50 = 9000 nM T20251 CWN90Q 54771978 IC50 = 32900 nM T20251 CUM4B5 54771980 IC50 = 7500 nM T20251 CL7UD5 54772203 IC50 = 16000 nM T20251 CH7K6J 54772204 IC50 = 12900 nM T20251 C4E5YQ 54772205 IC50 = 6600 nM T20251 C7Y8KR 54772206 IC50 = 20200 nM T20251 C8WHT5 56593934 IC50 = 7943.28 nM T20251 C8KO5T 56595054 IC50 = 720 nM T20251 CW89BT 56595402 IC50 > 10000 nM T20251 C4C3XQ 56595529 IC50 > 10000 nM T20251 CXEH21 56595883 IC50 > 10000 nM T20251 C7G4FQ 56596230 IC50 > 50000 nM T20251 CCG6D9 56597407 IC50 = 5500 nM T20251 CAC5B2 56597542 IC50 = 9800 nM T20251 CTK41N 56597689 IC50 = 8600 nM T20251 CN54TH 56597851 IC50 = 10000 nM T20251 CZNV53 56597988 IC50 = 15000 nM T20251 CI6B8D 56597990 IC50 > 33000 nM T20251 CSU5C1 56597991 IC50 > 33000 nM T20251 CJ4V0G 56598130 IC50 = 21000 nM T20251 CCR0Z1 56598517 IC50 > 25000 nM T20251 CK6VF3 56598528 IC50 = 8500 nM T20251 C91PGO 56603115 IC50 = 14700 nM T20251 C5ES6P 56603116 IC50 = 5400 nM T20251 CVI51O 56603118 IC50 = 19500 nM T20251 C2IM6T 56603174 IC50 = 4900 nM T20251 CH05TN 56603175 IC50 = 4400 nM T20251 CDL94H 56603301 IC50 = 1200 nM T20251 C9D1MV 56603353 IC50 = 16000 nM T20251 C60YTB 56603356 IC50 = 560 nM T20251 C9ZF6B 56643412 IC50 = 1200 nM T20251 CGX06Z 56643450 IC50 = 5000 nM T20251 CQ18BI 56643478 IC50 = 3700 nM T20251 CXI5V1 56643481 IC50 = 4840 nM T20251 CH3BN6 56643486 IC50 = 3460 nM T20251 CNB76L 56643505 IC50 > 30000 nM T20251 CS5P3M 56643544 IC50 = 24000 nM T20251 C6XI4W 56647652 IC50 = 4310 nM T20251 CUGA78 56649284 IC50 = 15500 nM T20251 C94RZF 56657929 IC50 = 10000 nM T20251 COST81 56657930 IC50 = 12000 nM T20251 CP2B8C 56657939 Ki = 5 nM T20251 CJ93HB 56657949 IC50 = 360 nM T20251 C13WTO 56658050 IC50 = 24000 nM T20251 C71XNV 56658572 IC50 = 2300 nM T20251 C21NEQ 56659196 IC50 > 50000 nM T20251 C7B9TW 56659197 IC50 = 25000 nM T20251 CL2YE8 56659224 IC50 = 4600 nM T20251 C5F1TD 56659225 IC50 = 10000 nM T20251 CUM53N 56659295 IC50 = 8.7 nM T20251 CVG04B 56659303 IC50 = 501.19 nM T20251 CRTE61 56659304 IC50 = 1000 nM T20251 C3R8ZJ 56659305 IC50 = 2511.89 nM T20251 CXBH95 56659572 Ki = 7200 nM T20251 CS4N2M 56659870 IC50 > 10000 nM T20251 CI1Z4B 56659871 IC50 = 8100 nM T20251 C0PSG1 56659872 IC50 = 2150 nM T20251 CJZS68 56660076 Ki = 27000 nM T20251 C4IZL5 56661444 IC50 = 4700 nM T20251 CQ25TB 56661451 IC50 = 18000 nM T20251 CM6A3K 56661468 Ki = 190 nM T20251 CC3XP8 56661559 IC50 = 25000 nM T20251 CCA76B 56661560 IC50 = 9400 nM T20251 C4H3VZ 56661561 IC50 = 17000 nM T20251 C43ICJ 56661679 IC50 = 4300 nM T20251 CJ0VW5 56662035 IC50 = 1300 nM T20251 CXFL76 56662692 IC50 > 33000 nM T20251 C7K4TJ 56662695 IC50 = 23000 nM T20251 CO3I1H 56662705 IC50 = 10000 nM T20251 CF45CH 56662780 IC50 = 4730 nM T20251 CP2LW0 56662936 IC50 = 316 nM T20251 CME1K7 56663526 Ki = 15000 nM T20251 CMI4D9 56663528 Ki = 12000 nM T20251 C9T2JQ 56663564 IC50 = 9900 nM T20251 C1KDU3 56663565 IC50 = 12000 nM T20251 CO1E6D 56663566 IC50 = 9400 nM T20251 CED2I5 56663567 IC50 = 4300 nM T20251 C3XW6G 56664901 Ki = 818 nM T20251 C9WDB6 56664902 IC50 = 8400 nM T20251 C7SJH2 56664979 IC50 = 840 nM T20251 CMY64U 56665506 IC50 = 45000 nM T20251 CL4XG3 56666171 IC50 = 7200 nM T20251 C6B7WR 56666236 IC50 = 2511.89 nM T20251 CVBA49 56666237 IC50 = 2511.89 nM T20251 C45XIM 56666238 IC50 > 50118.72 nM T20251 CHB63V 56666239 IC50 = 40000 nM T20251 CMZ6K8 56666240 IC50 = 8400 nM T20251 CYA27T 56666252 IC50 = 920 nM T20251 CL0BX9 56666253 IC50 = 310 nM T20251 C6I7DL 56666254 IC50 = 480 nM T20251 C0QOY7 56666255 IC50 = 2350 nM T20251 C4MFS5 56666758 IC50 = 320 nM T20251 CF0KZ2 56666759 IC50 > 10000 nM T20251 C62JDU 56666760 IC50 > 10000 nM T20251 CZG61M 56666868 IC50 = 4730 nM T20251 CLF45N 56666970 Ki > 29000 nM T20251 CUL0F4 56667010 IC50 = 8800 nM T20251 C9G1FY 56667011 IC50 = 14000 nM T20251 CA6K8E 56667012 IC50 = 8100 nM T20251 C2HXG3 56667013 IC50 = 1300 nM T20251 CC5S6K 56667036 IC50 = 3800 nM T20251 CF2N5W 56668309 IC50 = 12000 nM T20251 C4SP2W 56668313 IC50 = 4100 nM T20251 CT37LU 56668326 Ki = 13 nM T20251 C31SKP 56668413 IC50 > 50000 nM T20251 CJ95CA 56668427 Ki = 14 nM T20251 CX4Z9G 56668494 IC50 > 30000 nM T20251 CF7LR5 56668542 IC50 = 7100 nM T20251 CVGX27 56668837 Ki > 29000 nM T20251 CRVH74 56668949 IC50 > 100000 nM T20251 CKO8M6 56669554 IC50 > 33000 nM T20251 CI5Y4E 56669631 IC50 > 50 nM T20251 C5OF9G 56669642 IC50 = 3981.07 nM T20251 C4NR8W 56669644 IC50 = 16800 nM T20251 C5LE0N 56669662 IC50 = 1500 nM T20251 C36RHL 56669664 IC50 = 1570 nM T20251 C2HW9M 56669665 IC50 = 1900 nM T20251 CF06GH 56669910 Ki > 29000 nM T20251 CZO49F 56670192 IC50 = 2490 nM T20251 C5K4NS 56670257 IC50 = 8181.82 nM T20251 C9P6EQ 56670309 IC50 = 1500 nM T20251 CF23IK 56670310 IC50 = 4760 nM T20251 CRE51K 56670312 IC50 = 1570 nM T20251 CC7FH3 56670429 Ki = 1200 nM T20251 C76KFA 56670457 IC50 > 33000 nM T20251 C0I6AP 56670458 IC50 = 5300 nM T20251 C9Y8PV 56670459 IC50 = 10000 nM T20251 C5E7OB 56670460 IC50 = 16000 nM T20251 CCPY59 56670461 IC50 = 14000 nM T20251 CUP61N 56671791 IC50 = 1584.89 nM T20251 C34WPT 56671792 IC50 = 36000 nM T20251 CXUJ14 56671793 IC50 = 24000 nM T20251 C4UHW2 56671794 IC50 = 12000 nM T20251 CG1JX9 56671795 IC50 > 50000 nM T20251 CY0GX2 56671810 Ki = 10000 nM T20251 C2GFT1 56671811 Ki = 230 nM T20251 CCI1K3 56671812 Ki = 2220 nM T20251 C9GRW8 56671830 IC50 = 920 nM T20251 CXIQ98 56671923 IC50 = 1200 nM T20251 C19LWV 56671924 IC50 = 3100 nM T20251 CE3Y0C 56671925 IC50 = 8000 nM T20251 CX3LP4 56672008 IC50 = 22700 nM T20251 CET7K4 56672021 IC50 > 50 nM T20251 C29OYU 56672433 IC50 > 100000 nM T20251 CK9L4C 56672570 IC50 = 47300 nM T20251 CGAF01 56673075 IC50 = 14000 nM T20251 CP9Z2L 56673090 IC50 = 2000 nM T20251 C83MQK 56673091 IC50 = 2900 nM T20251 C6E7WM 56673153 IC50 = 794.33 nM T20251 C2Z1LP 56673154 IC50 = 3981.07 nM T20251 CC04NV 56673156 IC50 = 6000 nM T20251 C6FPR7 56673157 IC50 = 4800 nM T20251 C5G0ID 56673158 IC50 = 2480 nM T20251 C04ZUP 56673173 IC50 = 2800 nM T20251 C39ADI 56673420 Ki = 8400 nM T20251 C1E4CX 56673467 IC50 > 30000 nM T20251 C4G0YE 56673715 IC50 = 2190 nM T20251 CWZV47 56673716 IC50 = 390 nM T20251 C1KW9Z 56673717 IC50 = 5430 nM T20251 C19GOU 56673914 Ki = 17000 nM T20251 CW4J1Y 56673944 IC50 > 30000 nM T20251 CK5HP1 56673946 IC50 > 33000 nM T20251 C2D4JW 56673947 IC50 = 9400 nM T20251 CPU13M 56673948 IC50 = 4800 nM T20251 CY26SL 56675205 IC50 = 27000 nM T20251 CN3UM2 56675220 IC50 = 890 nM T20251 C03LOT 56675300 IC50 = 30000 nM T20251 CK9JX5 56675301 IC50 = 4500 nM T20251 CU0H6Z 56675302 IC50 = 7400 nM T20251 CJEA89 56675420 IC50 = 28000 nM T20251 C8JX6T 56675817 IC50 > 100000 nM T20251 CC73NZ 56676392 IC50 = 620 nM T20251 CP41OM 56676397 IC50 = 10000 nM T20251 CWS95P 56676398 IC50 = 5108.11 nM T20251 C0KG7I 56676474 IC50 = 11 nM T20251 CF3G7P 56676480 IC50 = 1584.89 nM T20251 CN4US8 56676481 IC50 = 3162.28 nM T20251 C49LUC 56676482 IC50 = 25118.86 nM T20251 CW86SU 56676730 Ki > 29000 nM T20251 CV79CF 56677248 Ki = 11000 nM T20251 CTW73X 56677275 IC50 = 1500 nM T20251 CHG64Z 56677276 IC50 = 9500 nM T20251 CBTG12 56677288 IC50 = 11700 nM T20251 CU35WX 56677289 IC50 = 7600 nM T20251 CE3T1U 56677296 IC50 = 1500 nM T20251 CP14LU 56678505 IC50 = 2511.89 nM T20251 CD8IZ5 56678506 IC50 = 25000 nM T20251 C7QW5F 56678507 IC50 = 44000 nM T20251 C7MXE5 56678508 IC50 = 27000 nM T20251 C5M0AS 56678518 Ki = 10000 nM T20251 C7IWP6 56678519 Ki = 1194 nM T20251 C0IGC6 56678520 Ki = 841 nM T20251 CT7BE0 56678521 Ki = 76 nM T20251 CUM2R9 56678534 IC50 = 160 nM T20251 C2O4SY 56678640 IC50 = 23000 nM T20251 CO9AX8 56678641 IC50 = 5800 nM T20251 C8QOB7 56678653 Ki = 90 nM T20251 CY5HJ2 56678654 Ki = 2747 nM T20251 CSHO51 56679737 IC50 = 10000 nM T20251 CDS09F 56679795 IC50 = 6309.57 nM T20251 CU04BI 56679796 IC50 = 7943.28 nM T20251 CTEK36 56679797 IC50 = 7943.28 nM T20251 COSK12 56679817 IC50 = 360 nM T20251 CM51TG 56679818 IC50 = 4980 nM T20251 CGCA84 56680098 IC50 > 30000 nM T20251 C9DTH0 56680351 IC50 = 1250 nM T20251 CMR0J9 56680352 IC50 > 10000 nM T20251 CDIZ56 56680456 IC50 = 3210 nM T20251 C67GMA 56680575 IC50 = 5100 nM T20251 C4MH8J 56681858 Ki = 1125 nM T20251 C1A0OH 56681872 IC50 = 130 nM T20251 C6ZOT4 56681873 IC50 = 460 nM T20251 C1XR6E 56681874 IC50 = 290 nM T20251 CPD15R 56681875 IC50 = 13830 nM T20251 C06HAF 56681960 IC50 = 38000 nM T20251 C1Y0MO 56682216 IC50 = 10000 nM T20251 CIW1T6 56683044 IC50 = 31000 nM T20251 CY1QA2 56683053 IC50 = 29000 nM T20251 C7F1JG 56683065 IC50 = 10000 nM T20251 CKVB12 56683116 IC50 = 17000 nM T20251 C9KMN5 56683121 IC50 = 16 nM T20251 CYJ1S0 56683143 IC50 = 3210 nM T20251 CBZG16 56683144 IC50 = 4760 nM T20251 CEYA71 56683146 IC50 = 1290 nM T20251 CP9G8Z 56683392 Ki > 29000 nM T20251 CR0E4M 56683440 IC50 > 30000 nM T20251 C4X7IP 56683681 IC50 = 2700 nM T20251 CIY31D 56683751 IC50 = 420 nM T20251 CH92EZ 56683889 Ki = 1700 nM T20251 CY1W2Q 56683890 Ki = 750 nM T20251 CWBF48 56683908 IC50 = 15000 nM T20251 C0MQ2W 56832511 IC50 = 16000 nM T20251 CE3PY9 56834574 IC50 = 23000 nM T20251 CD2FQ8 56834575 IC50 > 33000 nM T20251 CAJ3G0 56834577 IC50 = 206000 nM T20251 CY0K3F 56834578 IC50 > 33000 nM T20251 CMY23H 56834579 IC50 > 33000 nM T20251 CY92VU 56835087 IC50 > 30000 nM T20251 C0JMA7 56835088 IC50 = 7000 nM T20251 CR7LS4 56835090 IC50 = 20000 nM T20251 C4E6HV 56835171 Ki = 3235.94 nM T20251 CK7HJ8 56837192 Ki = 23000 nM T20251 C73MZW 56924689 IC50 = 13000 nM T20251 C8ZW3O 56927659 Ki = 1701 nM T20251 CV8W4T 56933229 IC50 > 300000 nM T20251 C9KI7Q 56940718 IC50 = 23700 nM T20251 CP5UD4 56944043 IC50 > 10000 nM T20251 C6F3VI 56944044 IC50 = 7700 nM T20251 C6GDX1 56944245 IC50 = 2200 nM T20251 CB0P9N 56944383 IC50 = 4000 nM T20251 C09WRF 56944429 IC50 = 4800 nM T20251 CHRU78 56946423 IC50 = 3300 nM T20251 CDK93W 56946894 IC50 > 100000 nM T20251 C5LJE8 56951456 IC50 > 30000 nM T20251 C6N0ZI 56951457 IC50 > 30000 nM T20251 CL90EM 56951458 IC50 > 30000 nM T20251 CD3V1J 56952775 IC50 = 2800 nM T20251 C8L7SJ 56952776 IC50 = 2540 nM T20251 CR9Q2E 56952777 IC50 = 2890 nM T20251 C0L4QG 56952778 IC50 = 670 nM T20251 CKMG86 56953069 IC50 = 920 nM T20251 C4V6ET 56953070 IC50 = 1480 nM T20251 CAK91L 56955954 IC50 = 17318 nM T20251 CP8H0D 56962365 IC50 = 5800 nM T20251 C1TR4E 56963091 Ki = 10700 nM T20251 C9L6FD 56963908 IC50 = 400 nM T20251 CKN0Z8 56964577 IC50 > 25000 nM T20251 C62OJE 56970264 IC50 = 27400 nM T20251 CJ6DK1 56970422 IC50 = 1600 nM T20251 C7S9ER 56970466 IC50 > 30000 nM T20251 CDH38V 56970630 IC50 = 3000 nM T20251 C67JVW 56970631 IC50 = 670 nM T20251 C4DMU9 56970632 IC50 = 1900 nM T20251 C3RBO8 56970861 IC50 = 430 nM T20251 CJ5O6Y 56970863 IC50 = 670 nM T20251 C1DN0L 56970864 IC50 = 470 nM T20251 CRF6L7 56971088 IC50 = 12 nM T20251 CQ5IH3 56971089 IC50 <= 1000 nM T20251 C9N0LO 56971556 IC50 = 31 nM T20251 CONA69 57065698 IC50 = 4660 nM T20251 CT67IO 57325589 IC50 > 25000 nM T20251 CV5CP4 57326678 IC50 = 6480 nM T20251 CVK5A3 57328247 IC50 = 100000 nM T20251 CQT5I3 57328465 IC50 = 8500 nM T20251 CY3B1Z 57330204 IC50 = 3600 nM T20251 CHN80L 57331188 IC50 = 12000 nM T20251 C4E1NK 57331209 IC50 = 1400 nM T20251 C8PWJ3 57331210 IC50 = 14000 nM T20251 C1E3WV 57331240 IC50 = 160 nM T20251 C4WI9O 57331241 IC50 = 1300 nM T20251 C68CPW 57331268 IC50 = 2700 nM T20251 CD0WM9 57331302 IC50 = 18000 nM T20251 CY0W1H 57331373 IC50 = 1300 nM T20251 CLB5K0 57331386 IC50 = 101700 nM T20251 CGUA26 57331668 IC50 = 17000 nM T20251 C64PSR 57331747 IC50 = 46000 nM T20251 CH30RG 57334102 IC50 = 159 nM T20251 C6DK4O 57334404 IC50 = 820 nM T20251 CD9I4N 57334553 IC50 = 1591 nM T20251 CXQ47N 57334707 IC50 = 226 nM T20251 CEG4N8 57334716 Ki = 470 nM T20251 C0UW5Z 57341142 EC50 = 4500 nM T20251 CS2FH5 57341143 EC50 = 5800 nM T20251 C2AUM9 57341144 EC50 > 30000 nM T20251 CX1FQ0 57341332 EC50 > 30000 nM T20251 CN3Y9D 57341333 EC50 > 30000 nM T20251 C3H1GV 57341334 EC50 = 27500 nM T20251 C0Z3JI 57341335 EC50 > 30000 nM T20251 C83DHY 57341336 EC50 > 30000 nM T20251 CDU9W0 57341337 EC50 > 30000 nM T20251 CL45WN 57345320 IC50 = 8920 nM T20251 CHE2I1 57345500 IC50 = 950 nM T20251 C63TFM 57345501 IC50 = 13300 nM T20251 C8KT2F 57345502 IC50 = 10000 nM T20251 CYZ1S5 57345568 IC50 = 326 nM T20251 CW4QD9 57345597 IC50 = 3200 nM T20251 CBQK82 57345598 IC50 = 16100 nM T20251 C3REK0 57345599 IC50 = 1288.25 nM T20251 CX49PE 57345600 IC50 = 1299.87 nM T20251 CD50GK 57345628 IC50 = 8900 nM T20251 COTF12 57382553 IC50 = 25700 nM T20251 CBF53W 57384005 IC50 = 5500 nM T20251 CF1OM2 57384006 IC50 > 40000 nM T20251 C8X5JG 57384039 IC50 = 8600 nM T20251 CV0GJ4 57384040 IC50 > 33000 nM T20251 C73XBL 57384077 Ki = 369 nM T20251 C34DJP 57384236 IC50 = 17000 nM T20251 CEOC15 57384237 IC50 = 720 nM T20251 CY50WC 57384238 IC50 = 4700 nM T20251 C7S0ZR 57384239 IC50 = 15000 nM T20251 C2XN1G 57384481 IC50 = 370 nM T20251 CR73IZ 57384482 IC50 = 650 nM T20251 CR2M5H 57384483 IC50 = 8500 nM T20251 CQ72HI 57384749 IC50 = 8900 nM T20251 C68KGE 57384750 IC50 = 7100 nM T20251 CQX8J0 57385070 IC50 > 300000 nM T20251 CPS89B 57385071 IC50 > 300000 nM T20251 CNU9C0 57385072 IC50 > 300000 nM T20251 CG5MT6 57385073 IC50 > 300000 nM T20251 CMC8H6 57386782 IC50 > 30000 nM T20251 CCT5D4 57386783 IC50 = 7000 nM T20251 CC30XZ 57386784 IC50 = 2400 nM T20251 C79BXP 57386785 IC50 > 60000 nM T20251 CM6DV7 57387028 IC50 = 5700 nM T20251 C0GS4F 57387282 IC50 = 12000 nM T20251 C0TL9C 57387283 IC50 = 8000 nM T20251 CRV2P5 57387539 IC50 = 1400 nM T20251 CAU3G9 57387540 IC50 = 7800 nM T20251 CL2AO8 57387541 IC50 = 23000 nM T20251 C0XWL8 57387542 IC50 = 16000 nM T20251 CC4DK0 57387775 IC50 = 2500 nM T20251 CSH7D9 57390216 IC50 = 5400 nM T20251 CLN2F8 57390217 IC50 = 11000 nM T20251 CM37LJ 57390221 Ki = 600 nM T20251 C58KFP 57390222 Ki = 900 nM T20251 CSCB73 57390223 Ki = 620 nM T20251 CVO05U 57390547 IC50 = 7900 nM T20251 CP8D5L 57390807 Ki = 43000 nM T20251 CDJC72 57390808 Ki = 24000 nM T20251 CE03ZS 57390809 Ki = 29000 nM T20251 CR8MW2 57391205 IC50 > 100000 nM T20251 CI9UT0 57391292 IC50 = 13489.63 nM T20251 C78LTO 57391294 IC50 = 1300 nM T20251 C2AR3V 57391609 IC50 = 900 nM T20251 CCA7D3 57391720 IC50 = 5800 nM T20251 C5QD2I 57391722 IC50 = 7900 nM T20251 CBEO41 57391765 IC50 > 30 nM T20251 CK9L1O 57391766 IC50 > 30 nM T20251 CN1Q4Y 57391767 IC50 > 30 nM T20251 CC53ND 57391768 IC50 > 30 nM T20251 CKPB03 57391802 IC50 = 2800 nM T20251 C8SW9E 57391803 IC50 = 4300 nM T20251 C5UWC6 57391804 IC50 = 9000 nM T20251 C78QEY 57391805 IC50 = 16900 nM T20251 CYAQ83 57391806 IC50 = 21700 nM T20251 CZ1EH9 57391826 IC50 = 33000 nM T20251 COL58X 57391831 IC50 = 12000 nM T20251 C6SGK0 57391843 Ki > 3000 nM T20251 C3MUQ4 57392006 IC50 = 15000 nM T20251 C4S7ET 57392007 IC50 = 18000 nM T20251 CT96ZS 57392011 Ki = 4500 nM T20251 CB6C4T 57392012 Ki = 910 nM T20251 CCZJ34 57392013 Ki = 1300 nM T20251 CP48ZB 57392014 Ki = 880 nM T20251 CHSW27 57392492 IC50 < 1000 nM T20251 CX89LJ 57392493 IC50 = 1300 nM T20251 C16PSG 57392623 Ki = 20000 nM T20251 CFM8E5 57392624 Ki = 8200 nM T20251 CGB71E 57393073 IC50 = 2398.83 nM T20251 CPQC75 57393451 IC50 = 7900 nM T20251 CJTY79 57393468 IC50 > 30000 nM T20251 CKS3X9 57393534 IC50 = 28200 nM T20251 CM2EH0 57393535 IC50 > 30000 nM T20251 CVO5M3 57393573 IC50 = 450 nM T20251 C9K0MG 57393724 IC50 = 13000 nM T20251 C2V7SB 57393725 IC50 > 33000 nM T20251 CH97QF 57393726 Ki = 460 nM T20251 CM80PV 57393727 Ki = 250 nM T20251 CJE1N0 57393728 Ki = 160 nM T20251 CWC2E8 57393729 Ki = 340 nM T20251 C13XZY 57394046 IC50 = 52000 nM T20251 C2XNP7 57394056 IC50 = 200000 nM T20251 C6D7UA 57394195 IC50 = 3900 nM T20251 CHA2Q7 57394339 Ki = 20000 nM T20251 CS8M9I 57394340 Ki = 1800 nM T20251 CLP4Z8 57394341 Ki = 12000 nM T20251 C8PWV4 57394342 Ki = 10000 nM T20251 C16OJD 57394343 Ki = 5700 nM T20251 C0AJM8 57394344 Ki = 55000 nM T20251 C6HR3Q 57394345 Ki = 47000 nM T20251 C0XDZ8 57394407 IC50 = 2600 nM T20251 CNOH63 57394711 IC50 > 100000 nM T20251 CRE41N 57394797 IC50 = 9400 nM T20251 CGV90O 57395178 IC50 = 3200 nM T20251 C9G6OJ 57395179 IC50 = 32000 nM T20251 CGR9F3 57395184 IC50 = 6500 nM T20251 CTG35L 57395190 IC50 > 30000 nM T20251 C3QCD9 57395216 IC50 > 30 nM T20251 C94MZO 57395217 IC50 > 30 nM T20251 CDIF34 57395218 IC50 > 30 nM T20251 C81ASJ 57395219 IC50 > 30 nM T20251 C5USX7 57395248 IC50 = 1600 nM T20251 CJ80BU 57395249 IC50 = 1800 nM T20251 CSO4Z0 57395278 IC50 = 1000 nM T20251 C01VOH 57395286 Ki = 2600 nM T20251 CB09IO 57395287 IC50 = 2300 nM T20251 C9CI3A 57395445 IC50 = 20000 nM T20251 CZ9G4Q 57395446 IC50 = 8700 nM T20251 C6SUR4 57395447 IC50 > 33000 nM T20251 C6VQ7I 57395454 Ki = 300 nM T20251 CFE6D4 57395455 Ki = 300 nM T20251 C0CGK5 57395838 IC50 = 3000 nM T20251 CHX4Z7 57396095 Ki = 19000 nM T20251 CRS39Y 57396096 Ki = 6400 nM T20251 CLEH95 57396097 Ki > 60000 nM T20251 C4NVE2 57396098 Ki = 12000 nM T20251 C7PT9Q 57396099 Ki = 22000 nM T20251 C23WQH 57396100 Ki = 7700 nM T20251 CTI36W 57396117 IC50 > 30000 nM T20251 C6HBG0 57396813 IC50 = 3300 nM T20251 CWU1I0 57396950 IC50 = 1200 nM T20251 CR41GU 57396951 IC50 > 32 nM T20251 C9YT0S 57396952 IC50 = 14000 nM T20251 CTH3P5 57396953 IC50 = 4000 nM T20251 C3L4ED 57396970 IC50 = 1000 nM T20251 CO37CB 57396999 IC50 > 30 nM T20251 C0P8KM 57397016 IC50 = 6700 nM T20251 CE85SV 57397017 IC50 = 4400 nM T20251 CYC1Q5 57397055 Ki > 3000 nM T20251 C25FTZ 57397056 IC50 = 900 nM T20251 C9W6IB 57397288 IC50 = 3600 nM T20251 CP0A2G 57397289 IC50 = 28000 nM T20251 CG8O2H 57397290 IC50 > 30000 nM T20251 CB7XV5 57397291 IC50 = 17000 nM T20251 C9WB0G 57397294 Ki = 1400 nM T20251 C7GJ6H 57397295 Ki = 1100 nM T20251 C7ML8N 57397296 Ki = 850 nM T20251 CLR02T 57397297 Ki = 8400 nM T20251 CEYO28 57397298 Ki = 710 nM T20251 CB20QV 57397299 Ki = 4400 nM T20251 CDQS63 57397589 IC50 = 25000 nM T20251 CNX73U 57397760 IC50 = 1100 nM T20251 CC8EV2 57397761 IC50 = 900 nM T20251 CH4Z3O 57397916 Ki = 7000 nM T20251 C9Y6KG 57397934 IC50 > 30000 nM T20251 CKDZ14 57398339 IC50 = 13598.78 nM T20251 CE5JQ8 57398341 IC50 = 128.82 nM T20251 C8Y4UJ 57398343 IC50 = 33113.11 nM T20251 CYO6T8 57398750 IC50 > 30 nM T20251 CSU2O9 57398779 IC50 = 1100 nM T20251 C5D0RB 57398829 Ki > 3000 nM T20251 CL4I6O 57398830 Ki > 3000 nM T20251 CSW1C3 57398976 IC50 = 9900 nM T20251 C0JIL8 57398977 IC50 = 13000 nM T20251 CH25BK 57398981 Ki = 1800 nM T20251 C4EY3H 57398982 Ki = 1400 nM T20251 CNY94K 57398983 Ki = 240 nM T20251 CG1D3L 57398984 Ki = 1100 nM T20251 C2J7GK 57398992 Ki = 360 nM T20251 CP8KQ7 57399426 IC50 = 12000 nM T20251 C4H6LZ 57399427 IC50 = 4700 nM T20251 CB42RN 57399556 Ki = 12000 nM T20251 CJO70A 57400003 IC50 = 129.99 nM T20251 CR09LY 57400127 IC50 = 5011.87 nM T20251 CK97BJ 57400372 IC50 = 25000 nM T20251 CA5KO3 57400374 IC50 = 25000 nM T20251 CDQ57A 57400458 IC50 = 1900 nM T20251 CED9C4 57400459 IC50 = 2000 nM T20251 CR0BU6 57400501 Ki > 3000 nM T20251 CE82XL 57400502 IC50 = 2100 nM T20251 CWZ50O 57400503 IC50 = 930 nM T20251 CJBU02 57400505 IC50 = 1500 nM T20251 CH13FG 57400694 IC50 = 11000 nM T20251 C6W1SD 57400695 IC50 = 7300 nM T20251 C9IXS8 57400698 Ki = 900 nM T20251 CS0E7F 57401040 IC50 = 113000 nM T20251 CCL98E 57401058 IC50 = 29500 nM T20251 CU2V1C 57401137 IC50 = 15000 nM T20251 CVXU49 57401184 IC50 = 3000 nM T20251 CUYK04 57401306 Ki = 24000 nM T20251 CSQK78 57401307 Ki = 9300 nM T20251 C8GC4D 57401308 Ki = 7600 nM T20251 CFL71K 57401309 Ki = 13000 nM T20251 CJQ89O 57401397 Ki = 2100 nM T20251 CKA34L 57401798 IC50 = 3090.3 nM T20251 CF0CA4 57401801 IC50 = 33113.11 nM T20251 C9X7PT 57401860 IC50 = 6 nM T20251 C3EV5S 57401884 IC50 = 25100 nM T20251 CG0DR6 57402003 IC50 = 330 nM T20251 C5NDS6 57402175 IC50 = 3200 nM T20251 C7CG1T 57402187 IC50 > 30000 nM T20251 CV54BI 57402219 IC50 = 13200 nM T20251 CV2ME6 57402260 IC50 = 5000 nM T20251 CQ1A8P 57402261 IC50 = 1300 nM T20251 CW94QA 57402262 IC50 = 1800 nM T20251 CMJA69 57402263 IC50 = 3400 nM T20251 C5X0LN 57402288 IC50 = 16000 nM T20251 C9D3ZE 57402314 Ki > 3000 nM T20251 CXT2L1 57402315 IC50 = 3400 nM T20251 CJ0E6V 57402465 IC50 = 11000 nM T20251 C6PM9O 57402466 IC50 > 33000 nM T20251 C1G3WE 57402816 IC50 = 63100 nM T20251 C2WT8S 57402817 IC50 = 4900 nM T20251 C65TPY 57403054 IC50 = 27000 nM T20251 CQ1ZV2 57403067 Ki = 11000 nM T20251 CHA41T 57403138 IC50 = 25000 nM T20251 CO94YE 57403139 IC50 = 18000 nM T20251 CX94UQ 57403171 IC50 = 80000 nM T20251 CC0D8X 57403932 IC50 = 35000 nM T20251 CX31VN 57403989 IC50 = 12000 nM T20251 C49JDH 57404030 Ki > 10000 nM T20251 C9SB1D 57404031 Ki > 3000 nM T20251 C1L8YD 57404359 IC50 = 8800 nM T20251 C8SX7A 57404360 IC50 = 6100 nM T20251 C6WU8O 57406717 IC50 = 15000 nM T20251 C0M6NB 57406720 IC50 = 2700 nM T20251 CWCY97 57406911 IC50 > 33000 nM T20251 C5CRJ1 57412107 IC50 = 2380 nM T20251 CUSO25 57414544 IC50 = 62 nM T20251 C8UMR2 57414545 IC50 = 580 nM T20251 CSA3P9 57414546 IC50 = 39.81 nM T20251 CI2TO3 57414547 IC50 = 2.512 nM T20251 CA8K1N 57414548 IC50 = 7860 nM T20251 CX6N9E 57414549 IC50 = 192 nM T20251 C1CUJ7 57441855 IC50 = 4000 nM T20251 CF9Z3R 57441946 IC50 > 32000 nM T20251 CRV53F 57441994 IC50 > 32000 nM T20251 C47QNO 57442001 IC50 = 13200 nM T20251 CR58EY 57442010 IC50 > 32000 nM T20251 C54JSK 57448273 IC50 > 10000 nM T20251 CVNR58 57448274 IC50 = 2500 nM T20251 C5CBG4 57448276 IC50 = 2800 nM T20251 CUWK92 57448281 IC50 > 10000 nM T20251 CY86DR 57448284 IC50 = 8900 nM T20251 C74GKR 57448289 IC50 > 10000 nM T20251 CAE6B5 57448332 IC50 > 10000 nM T20251 CK9TD7 57448346 IC50 > 10000 nM T20251 CA6YR3 57448356 IC50 > 10000 nM T20251 C0I1CB 57448358 IC50 > 10000 nM T20251 CWA9F6 57482815 IC50 = 63095.73 nM T20251 C2QS1Y 57504248 IC50 = 50118.72 nM T20251 CMB2W7 57504266 IC50 = 19952.62 nM T20251 CAY71X 57504268 IC50 > 33000 nM T20251 CBU6N2 57504311 IC50 > 100000 nM T20251 C6S8CV 57504312 IC50 > 79432.82 nM T20251 C0W5QD 57504313 IC50 > 100000 nM T20251 CD85MW 57504320 IC50 = 31622.78 nM T20251 CH79YV 57504325 IC50 = 79432.82 nM T20251 CZ8SF5 57504326 IC50 = 63095.73 nM T20251 CRC5O1 57504327 IC50 = 15848.93 nM T20251 C7JDH2 57504328 IC50 = 50118.72 nM T20251 CM8Z6N 57504345 IC50 = 25118.86 nM T20251 CKE12J 57504346 IC50 = 12589.25 nM T20251 C4UAZ5 57504347 IC50 = 15848.93 nM T20251 CH3Y9K 57504348 IC50 = 63095.73 nM T20251 C9TY4W 57504354 IC50 = 19952.62 nM T20251 CCT08G 57504355 IC50 = 63095.73 nM T20251 C0OIW2 57504356 IC50 > 100000 nM T20251 CPQA09 57504358 IC50 = 10000 nM T20251 CP7BL3 57504360 IC50 = 63095.73 nM T20251 CV20RS 57504361 IC50 = 50118.72 nM T20251 C42OWY 57504362 IC50 > 100000 nM T20251 C8K7TB 57504363 IC50 = 79432.82 nM T20251 CPR02A 57504388 IC50 = 50118.72 nM T20251 CI74AT 57504389 IC50 = 50118.72 nM T20251 COB73U 57504402 IC50 = 15848.93 nM T20251 CLWU10 57504418 IC50 = 63095.73 nM T20251 C8UHW1 57504419 IC50 > 100000 nM T20251 C0BGQ4 57504420 IC50 > 100000 nM T20251 C38YSV 57504421 IC50 > 100000 nM T20251 C1CPF8 57504444 IC50 = 79432.82 nM T20251 CB54GY 57504445 IC50 = 10000 nM T20251 CYHT79 57504446 IC50 = 7943.28 nM T20251 CAV2N7 57504447 IC50 > 100000 nM T20251 C3AOX7 57504450 IC50 = 25118.86 nM T20251 CR0HE5 57504454 IC50 = 6309.57 nM T20251 CV8B0T 57504457 IC50 = 63095.73 nM T20251 CRLJ46 57504462 IC50 > 100000 nM T20251 CNEB25 57504463 IC50 = 31622.78 nM T20251 CR1A8Z 57504467 IC50 = 39810.72 nM T20251 C90OLN 57504474 IC50 = 26000 nM T20251 CB47MQ 57514846 IC50 > 10000 nM T20251 C7I4QD 57519510 IC50 > 30000 nM T20251 C3N4MF 57520842 IC50 > 30000 nM T20251 CEL56T 57520942 IC50 > 30000 nM T20251 C7PLG5 57521314 IC50 = 49800 nM T20251 CWE9J4 57522010 IC50 > 30000 nM T20251 C3I5XK 57522013 IC50 = 21900 nM T20251 C53BGU 57522014 IC50 > 30000 nM T20251 CHU5T7 57523687 IC50 = 27000 nM T20251 C5P3HT 57545640 Ki = 2314 nM T20251 CR34CL 57582353 IC50 > 30000 nM T20251 C7D1JL 57606048 IC50 = 105000 nM T20251 C9I6RO 57606050 IC50 > 33000 nM T20251 C6D3MG 57606067 IC50 > 33000 nM T20251 C3OQ4Z 57606068 IC50 > 33000 nM T20251 CYEQ10 57606070 IC50 > 33000 nM T20251 CY59ML 57606091 IC50 > 33000 nM T20251 C1F2DJ 57606095 IC50 > 33000 nM T20251 CI59LU 57609886 Ki = 498 nM T20251 C6GCQ8 57611057 IC50 = 9100 nM T20251 CYV5K2 57639150 IC50 = 38100 nM T20251 CM32RA 57656640 IC50 = 7100 nM T20251 C0OJA5 57656641 IC50 = 6300 nM T20251 CT8V9X 57656657 IC50 = 890 nM T20251 CH7BO0 57656701 IC50 = 13000 nM T20251 CMI4T3 57656713 IC50 = 400 nM T20251 CB30PQ 57656715 IC50 = 2000 nM T20251 C51DOT 57656719 IC50 = 6300 nM T20251 C2GHC7 57656729 IC50 = 5000 nM T20251 C6W3EJ 57656749 IC50 = 6300 nM T20251 C1KAC6 57656808 IC50 = 8900 nM T20251 CN7O1T 57656825 IC50 = 14000 nM T20251 CHJ87A 57656833 IC50 = 60000 nM T20251 CS6O1V 57656854 IC50 = 19000 nM T20251 CPN5S4 57656869 IC50 = 16000 nM T20251 CU8I2F 57656871 IC50 = 10000 nM T20251 CD5W4E 57656887 IC50 = 28000 nM T20251 CQX1D5 57656921 IC50 = 7100 nM T20251 C1QSF4 57656938 IC50 = 13000 nM T20251 C5V0JI 57656942 IC50 = 14000 nM T20251 CJYS25 57663369 IC50 = 7943.28 nM T20251 C4QG8R 57663382 IC50 = 6309.57 nM T20251 CHQI67 57663405 IC50 > 63095.73 nM T20251 CA9RK8 57663418 IC50 = 7943.28 nM T20251 CM7H9G 57663419 IC50 = 19952.62 nM T20251 C58ERT 57663421 IC50 = 15848.93 nM T20251 CY2S7K 57663434 IC50 = 1995.26 nM T20251 C9A0XM 57663447 IC50 = 25118.86 nM T20251 C18FHN 57663450 IC50 = 12589.25 nM T20251 CPSX03 57663451 IC50 = 7943.28 nM T20251 CMUD63 57663495 IC50 = 12589.25 nM T20251 CVL35Z 57663496 IC50 = 19952.62 nM T20251 CBK0Y1 57663581 IC50 = 63095.73 nM T20251 CSK82C 57663586 IC50 = 15848.93 nM T20251 C5J1QT 57663596 IC50 = 29512.09 nM T20251 CTV29J 57663598 IC50 = 19952.62 nM T20251 C2X7OT 57663610 IC50 = 12589.25 nM T20251 C98CVM 57663630 IC50 = 15848.93 nM T20251 CGA1V2 57663637 IC50 > 63095.73 nM T20251 CV2J9A 57663655 IC50 = 18620.87 nM T20251 CR7S5U 57663666 IC50 = 19952.62 nM T20251 C4GXF1 57663688 IC50 = 12589.25 nM T20251 CZ2UB5 57705473 IC50 > 10000 nM T20251 C35GXV 57720515 EC50 = 6000 nM T20251 CQP7E0 57750290 IC50 = 21030 nM T20251 C1U3YR 57750299 IC50 > 33300 nM T20251 CEY8W0 57750311 IC50 > 33300 nM T20251 CNBO65 57750312 IC50 = 80124 nM T20251 C2F9DS 57750315 IC50 > 100000 nM T20251 CZ08KN 57750321 IC50 > 100000 nM T20251 CUY8T6 57750329 IC50 > 33300 nM T20251 CK4W1L 57750342 IC50 > 33300 nM T20251 CM5X9L 57750343 IC50 = 9092 nM T20251 C0TNP8 57750364 IC50 > 33300 nM T20251 CBY5E4 57750369 IC50 = 74807 nM T20251 CO6P5G 57750381 IC50 > 33300 nM T20251 CSI9Y4 57750382 IC50 = 1600 nM T20251 C6GH7X 57750391 IC50 = 3500 nM T20251 CL7CW0 57750402 IC50 = 9369 nM T20251 CA4G5W 57750407 IC50 = 29367 nM T20251 CM7XL6 57750408 IC50 = 6747 nM T20251 CY4Z8R 57750418 IC50 = 26957 nM T20251 C8OY4I 57750420 IC50 > 33300 nM T20251 CT89JH 57780007 IC50 = 50118.72 nM T20251 CT8RO7 57780008 IC50 = 7943.28 nM T20251 C5RIN4 57780016 IC50 > 63095.73 nM T20251 CE9WC0 57780017 IC50 = 15848.93 nM T20251 C1W4SB 57780018 IC50 = 31622.78 nM T20251 CT96WD 57780020 IC50 = 2511.89 nM T20251 C9FH4B 57790981 IC50 = 5500 nM T20251 CG16CV 57916503 IC50 > 100000 nM T20251 C8E6PG 57927934 IC50 > 33000 nM T20251 C10VYA 57948490 IC50 > 30000 nM T20251 CAU57Q 57969602 IC50 = 3000 nM T20251 C1LZI4 57969746 IC50 > 10000 nM T20251 CXI6A1 57970302 IC50 = 1000 nM T20251 C67MSZ 58017509 IC50 = 14000 nM T20251 CG9V4E 58017514 IC50 = 15000 nM T20251 CN6Z0X 58017523 IC50 = 5600 nM T20251 C7M3DS 58017531 IC50 > 33000 nM T20251 C1EP6I 58024825 IC50 > 29000 nM T20251 C19XQV 58026164 IC50 = 20000 nM T20251 CEWR70 58065681 IC50 = 5200 nM T20251 C9JCL7 58080768 IC50 = 4900 nM T20251 C5B0RJ 58083331 Ki = 33600 nM T20251 C1C6OS 58083336 Ki = 31200 nM T20251 C6DZ0X 58083358 Ki = 23000 nM T20251 CND4G1 58088117 IC50 = 2500 nM T20251 C2EY8P 58109378 IC50 = 5300 nM T20251 CJ07OW 58109450 IC50 = 6300 nM T20251 C4FH0W 58118983 IC50 > 10000 nM T20251 C46AUK 58137055 IC50 > 32000 nM T20251 C7ONC3 58137106 IC50 > 33000 nM T20251 CRPL37 58137176 IC50 > 32000 nM T20251 C2R3IZ 58178960 IC50 = 7200 nM T20251 C1TL8P 58179284 IC50 > 30000 nM T20251 C7AY1J 58190324 IC50 = 11000 nM T20251 CI63UA 58190330 IC50 > 30000 nM T20251 CPQ0Z4 58269588 IC50 > 30000 nM T20251 CD18IU 58269609 IC50 > 30000 nM T20251 C8ILS3 58269629 IC50 = 27000 nM T20251 C5VFQ7 58269655 IC50 = 4000 nM T20251 C2PYB1 58269668 IC50 > 30000 nM T20251 C3CFB8 58269691 IC50 > 30000 nM T20251 CTWG72 58290872 IC50 = 24500 nM T20251 CJ4B6P 58299601 IC50 = 2000 nM T20251 CT78UE 58299836 IC50 = 720 nM T20251 CB3IT1 58302173 Ki > 30000 nM T20251 CW1G9J 58302348 Ki = 740 nM T20251 C0F3BO 58394783 IC50 > 100000 nM T20251 C0X7IK 58394837 IC50 > 100000 nM T20251 CASI81 58395078 IC50 > 100000 nM T20251 CWBM72 58395283 IC50 = 20000 nM T20251 CZ2VK4 58408526 Ki = 8820 nM T20251 CE80UP 58438175 IC50 > 30000 nM T20251 C5DC7T 58438322 IC50 = 1300 nM T20251 C9UK7P 58438475 IC50 = 2900 nM T20251 CC8TK0 58466119 Ki > 10000 nM T20251 C9IRW0 58466120 Ki > 15000 nM T20251 CSU91B 58466122 Ki > 15000 nM T20251 CKSF73 58466243 Ki = 1240 nM T20251 CH9ER4 58466295 Ki = 6900 nM T20251 C6QJX4 58466300 Ki > 10000 nM T20251 C6OJC2 58466301 Ki = 496 nM T20251 CBN9L0 58561169 IC50 = 600 nM T20251 CIJ09G 58576126 IC50 = 58 nM T20251 C4VT6Z 58615686 IC50 = 3180 nM T20251 C6JKM0 58834906 IC50 = 9900 nM T20251 CF9Z0L 58834953 IC50 = 18000 nM T20251 C4PWA9 58835024 IC50 > 30000 nM T20251 CCR4T7 58835217 IC50 > 30000 nM T20251 C9ZE7J 58874273 IC50 > 10000 nM T20251 CCNI49 58920310 IC50 = 22000 nM T20251 CXGW57 58920485 IC50 > 80000 nM T20251 CETS76 59019389 IC50 > 16000 nM T20251 CJS46Y 59086459 IC50 = 7300 nM T20251 CO6TL1 59135478 IC50 = 420 nM T20251 C31KUT 59149763 IC50 = 11220.18 nM T20251 CH41MU 59149828 IC50 > 100000 nM T20251 CCQM76 59153288 IC50 > 30000 nM T20251 C0Z5IL 59173801 IC50 = 3080 nM T20251 CWJT87 59174010 IC50 = 1290 nM T20251 C3L4JY 59176329 IC50 = 3900 nM T20251 CW24YS 59190451 IC50 = 6309.57 nM T20251 CEI8A5 59190544 IC50 = 19952.62 nM T20251 CY54RB 59199467 IC50 = 4800 nM T20251 C94HKZ 59199478 IC50 = 1700 nM T20251 CMSR93 59199482 IC50 = 6300 nM T20251 C30VAF 59199488 IC50 = 3500 nM T20251 CNUT13 59218182 IC50 > 10000 nM T20251 CHVU94 59218184 IC50 > 10000 nM T20251 CY6EB4 59218190 IC50 > 10000 nM T20251 C2PJ4N 59271992 IC50 = 13000 nM T20251 C7XM1P 59272333 Ki > 15000 nM T20251 CWCK45 59272335 Ki = 14000 nM T20251 C9VNB7 59275242 IC50 = 5800 nM T20251 CTF1U6 59275404 IC50 = 18000 nM T20251 C4KU2S 59278286 IC50 > 30000 nM T20251 CEAY32 59278314 IC50 = 30000 nM T20251 CN1Y9X 59279548 IC50 = 39810.72 nM T20251 CC1AN4 59279550 IC50 = 12589.25 nM T20251 CM4XB0 59279551 IC50 = 39810.72 nM T20251 CBWJ84 59291203 IC50 > 33000 nM T20251 CPWM60 59291925 IC50 > 100000 nM T20251 CE6KO4 59291951 IC50 > 100000 nM T20251 CT3EW2 59292007 IC50 > 100000 nM T20251 C2PE0T 59292008 IC50 > 100000 nM T20251 C90EAP 59295914 IC50 = 3162.28 nM T20251 CFX9H8 59295925 IC50 = 6309.57 nM T20251 C5P6UI 59295926 IC50 = 6309.57 nM T20251 C18YQX 59295928 IC50 > 31622.78 nM T20251 C9NMZ2 59295931 IC50 = 251.19 nM T20251 CA8T3Q 59295938 IC50 = 5011.87 nM T20251 C59QBR 59295939 IC50 = 1995.26 nM T20251 COG4S6 59295946 IC50 = 5011.87 nM T20251 CHP65R 59295958 IC50 = 1258.93 nM T20251 C3PCY5 59295968 IC50 > 31622.78 nM T20251 CYG56K 59295969 IC50 = 794.33 nM T20251 C4PYU5 59295974 IC50 > 31622.78 nM T20251 CRZN12 59295978 IC50 = 1995.26 nM T20251 CR2T5D 59295982 IC50 > 6309.57 nM T20251 C17USX 59295994 IC50 > 10000 nM T20251 CJV58T 59296000 IC50 = 501.19 nM T20251 C2K1TV 59296010 IC50 = 398.11 nM T20251 C0KM5W 59296024 IC50 > 31622.78 nM T20251 CE73NG 59296033 IC50 = 1000 nM T20251 CT2P4Z 59296039 IC50 = 251.19 nM T20251 CXK7O5 59296048 IC50 = 1995.26 nM T20251 CPE0B2 59296066 IC50 = 10000 nM T20251 CFR8S7 59296077 IC50 = 1995.26 nM T20251 CMD56H 59296081 IC50 = 1000 nM T20251 CFCE90 59296090 IC50 = 5011.87 nM T20251 CUC57E 59296099 IC50 = 1995.26 nM T20251 C1ZN0M 59296100 IC50 = 1258.93 nM T20251 CX6JS1 59296104 IC50 = 1995.26 nM T20251 C5TMB2 59296111 IC50 = 3162.28 nM T20251 C6E5UG 59366166 Ki < 13 nM T20251 CSF3A7 59394005 IC50 = 7000 nM T20251 CP34RY 59394193 IC50 > 30000 nM T20251 C5IQ4P 59394335 IC50 = 23500 nM T20251 CY9RB5 59394429 IC50 = 15600 nM T20251 CHXC24 59394467 IC50 = 11100 nM T20251 C7A5KZ 59394725 IC50 = 7400 nM T20251 CK4Y8T 59395224 IC50 > 33000 nM T20251 CDA17U 59396249 IC50 = 46100 nM T20251 C80HTM 59396252 IC50 = 78600 nM T20251 CE01DO 59396594 IC50 = 76000 nM T20251 C6IDV0 59396641 IC50 = 50100 nM T20251 CQK9S3 59401826 IC50 = 1000 nM T20251 C53BVH 59401876 IC50 = 480 nM T20251 CNOI48 59401886 IC50 = 1800 nM T20251 C29YCJ 59411406 IC50 = 27100 nM T20251 C03EFU 59440893 IC50 > 30000 nM T20251 CPUZ69 59447115 IC50 > 10000 nM T20251 CK6LX0 59454220 IC50 = 7000 nM T20251 C2SDN1 59454252 IC50 = 5000 nM T20251 C46UHJ 59458228 IC50 = 33000 nM T20251 CSOL31 59458454 IC50 > 80000 nM T20251 C0L2FW 59458459 IC50 = 44000 nM T20251 C83DOJ 59458460 IC50 = 11000 nM T20251 C0ZLU4 59458594 IC50 = 23000 nM T20251 CZ0Q7W 59458647 IC50 > 80000 nM T20251 CV41DL 59458714 IC50 > 80000 nM T20251 C6K0MO 59458732 IC50 = 21000 nM T20251 CFP75N 59458738 IC50 = 16000 nM T20251 CJ5I3Q 59459021 IC50 = 25600 nM T20251 C9XI4D 59459390 IC50 = 63000 nM T20251 CTH04J 59459492 IC50 = 12000 nM T20251 C1E3XT 59472470 EC50 = 15000 nM T20251 C92NPY 59472493 IC50 = 18100 nM T20251 CL4F1U 59472507 IC50 = 800 nM T20251 CG1ZH6 59472511 IC50 = 1580 nM T20251 CHU2S4 59472516 IC50 = 1390 nM T20251 CW4I0H 59472517 IC50 = 2680 nM T20251 C4RZ7E 59472522 IC50 = 17600 nM T20251 CKS31U 59472524 IC50 = 8740 nM T20251 C35EKB 59472530 IC50 = 530 nM T20251 CLB40A 59472544 EC50 = 1300 nM T20251 CL9Y0P 59472546 IC50 = 4030 nM T20251 CXH19J 59472574 IC50 = 2610 nM T20251 C51KUS 59472588 IC50 = 3560 nM T20251 CS87XI 59472603 IC50 = 8960 nM T20251 CI8H4T 59472630 IC50 = 3050 nM T20251 CXO21N 59472637 IC50 = 20800 nM T20251 CH0S6A 59472641 IC50 = 4060 nM T20251 C0LBN5 59472644 IC50 > 10000 nM T20251 C4SR9V 59472646 IC50 > 30000 nM T20251 C6D7LS 59472679 IC50 = 3680 nM T20251 C8UMR6 59472684 IC50 = 1830 nM T20251 C1ME7D 59472698 IC50 = 1010 nM T20251 CYO06N 59472699 IC50 = 870 nM T20251 C6XDH2 59472707 IC50 = 800 nM T20251 CF72WU 59472713 IC50 = 3220 nM T20251 C9L0GJ 59472717 IC50 = 43900 nM T20251 CJR3K7 59472756 IC50 = 1490 nM T20251 C1RUN6 59472765 Ki = 3600 nM T20251 CZ52KP 59472771 IC50 = 10300 nM T20251 CB3X0F 59472773 IC50 = 7570 nM T20251 C6YZR8 59472775 IC50 = 44200 nM T20251 CDOV85 59472789 IC50 > 30000 nM T20251 CWD0K3 59472815 IC50 = 2870 nM T20251 C15JGP 59472849 IC50 = 6220 nM T20251 CM0G7S 59472858 IC50 > 50000 nM T20251 CEP94I 59472861 IC50 = 630 nM T20251 CLH47W 59472872 IC50 = 2220 nM T20251 C2SNL8 59541239 IC50 = 12000 nM T20251 CA9NE4 59548712 IC50 = 8000 nM T20251 CG2V1M 59568650 IC50 = 14000 nM T20251 C7FAN1 59568652 IC50 = 18000 nM T20251 CM1G2P 59568656 IC50 = 33000 nM T20251 CS19JW 59568702 IC50 = 22000 nM T20251 C4W8RH 59651989 IC50 > 30000 nM T20251 CIL17E 59652016 IC50 = 18000 nM T20251 CF8E1J 59764390 IC50 = 400 nM T20251 CC48EN 59764418 IC50 = 5300 nM T20251 C4NBG7 59764433 IC50 = 3020 nM T20251 C40UZT 59764460 IC50 = 2640 nM T20251 C6AQX8 59764524 IC50 = 3350 nM T20251 CJ7E6C 60026483 IC50 = 3800 nM T20251 C45XVN 60142198 Ki = 1980 nM T20251 CJ5M9S 60142200 Ki = 1740 nM T20251 C79ZOY 60142335 Ki = 4800 nM T20251 CNKF60 60143411 IC50 = 27600 nM T20251 CYCN68 60143412 IC50 > 100000 nM T20251 CJP6A3 60143413 IC50 > 100000 nM T20251 CX9PB5 60143414 IC50 > 100000 nM T20251 CGJ5H3 60143415 IC50 > 100000 nM T20251 C7TC5K 60143416 IC50 > 100000 nM T20251 CRFV62 60143588 IC50 > 100000 nM T20251 C7S4PH 60143589 IC50 > 100000 nM T20251 C9EH3R 60143590 IC50 = 78700 nM T20251 CZ3QD9 60143591 IC50 > 100000 nM T20251 CM62NL 60143592 IC50 > 100000 nM T20251 C9ME8V 60143757 IC50 > 100000 nM T20251 CFH4L9 60143758 IC50 > 100000 nM T20251 C4R6PH 60143759 IC50 = 49100 nM T20251 CVA2X8 60143760 IC50 > 100000 nM T20251 CD65CK 60143761 IC50 > 100000 nM T20251 C4TES3 60143762 IC50 > 100000 nM T20251 CR1ZN4 60143921 IC50 > 100000 nM T20251 CD5T7O 60143922 IC50 > 100000 nM T20251 C5DJA6 60143923 IC50 > 100000 nM T20251 CPF6A9 60143924 IC50 > 100000 nM T20251 CRTN28 60143925 IC50 > 100000 nM T20251 CYJ19Q 60143926 IC50 > 100000 nM T20251 C8UQ7D 60144084 IC50 > 100000 nM T20251 CM0C9O 60144086 IC50 > 100000 nM T20251 CN4A8W 60144088 IC50 > 100000 nM T20251 CJ4XM3 60144089 IC50 > 100000 nM T20251 CY4H9Z 60144244 IC50 > 100000 nM T20251 CMQ78O 60144245 IC50 > 100000 nM T20251 CAPO85 60145490 IC50 = 76500 nM T20251 C4KZ3M 60145492 IC50 > 100000 nM T20251 CBP2K4 60145493 IC50 = 13600 nM T20251 C0B7QX 60145494 IC50 = 18800 nM T20251 CDK1O7 60145629 IC50 > 100000 nM T20251 COR56Z 60145630 IC50 > 100000 nM T20251 C03HNY 60145631 IC50 > 100000 nM T20251 C6CE5G 60145632 IC50 > 100000 nM T20251 CJSV45 60145633 IC50 > 100000 nM T20251 CB4ND5 60145634 IC50 = 26100 nM T20251 C0FR9I 60145771 IC50 > 100000 nM T20251 C8S4EL 60145772 IC50 > 100000 nM T20251 CE17ZH 60145773 IC50 > 100000 nM T20251 CHJ03O 60145774 IC50 > 100000 nM T20251 C40GSO 60145775 IC50 > 100000 nM T20251 CQW7A8 60149247 IC50 = 9000 nM T20251 CGF54X 60150483 IC50 = 5600 nM T20251 C3HZ5J 60150507 IC50 = 2500 nM T20251 C30UIB 60150707 IC50 = 5400 nM T20251 CTL97W 60151476 IC50 > 10000 nM T20251 C3D2ZI 60155056 IC50 > 24000 nM T20251 CA4OH9 60155057 IC50 > 23400 nM T20251 CR36EQ 60155058 IC50 > 22700 nM T20251 CT7ID2 60162269 IC50 = 8240 nM T20251 C2D3HQ 60168069 IC50 = 73600 nM T20251 CSN5C8 60170856 IC50 > 10000 nM T20251 CPLU74 60170970 IC50 = 9700 nM T20251 C6U0HA 60194465 IC50 = 14500 nM T20251 CYH8P0 60199250 IC50 > 30000 nM T20251 C4VZ5L 60199310 IC50 = 23990 nM T20251 CSPU20 60199433 IC50 > 30000 nM T20251 CEKA47 60199634 IC50 = 15000 nM T20251 CC8YH1 60199796 IC50 = 75000 nM T20251 C2TY3G 60199965 IC50 = 168000 nM T20251 CR4IL3 60199967 IC50 = 25000 nM T20251 CPK52S 60200126 IC50 = 32000 nM T20251 C29HIU 60200128 IC50 > 333000 nM T20251 COJ18I 60200280 IC50 = 152000 nM T20251 CO5HD0 60201085 IC50 = 5300 nM T20251 CA57OQ 60201086 IC50 = 4900 nM T20251 C5UKQ8 60201087 IC50 = 11000 nM T20251 CA7NI3 60201088 IC50 = 24000 nM T20251 C1YQ8J 60201256 IC50 > 33000 nM T20251 CM92ST 60201265 IC50 = 189000 nM T20251 C5WQ3Z 60201425 IC50 = 88000 nM T20251 CN18KX 60201945 IC50 = 199000 nM T20251 CJ23UN 60201946 IC50 = 57000 nM T20251 C6Z2HF 60201948 IC50 = 75000 nM T20251 C2D0TI 60202105 IC50 = 156000 nM T20251 CK3G6T 60202107 IC50 = 117000 nM T20251 CY04QB 60210882 IC50 > 10000 nM T20251 CL42CH 60509567 IC50 = 0.76 nM T20251 CW3H0V 60634975 IC50 > 25000 nM T20251 C4BZ2N 60637368 IC50 < 10000 nM T20251 CI7DY2 60965486 IC50 > 10000 nM T20251 C02TAQ 62705172 IC50 > 50000 nM T20251 CV0X4K 62705173 IC50 > 50000 nM T20251 CG2VD0 62705174 IC50 > 50000 nM T20251 CWL9J4 62705175 IC50 = 6300 nM T20251 CQ5LS1 62705176 IC50 = 6600 nM T20251 CK2DG6 62705177 IC50 = 9300 nM T20251 CX7Q2A 62705299 IC50 > 10000 nM T20251 C59QUB 62705330 IC50 = 13000 nM T20251 CANL67 62705331 IC50 > 50000 nM T20251 CW19CI 62705332 IC50 = 46000 nM T20251 CK2WS1 62705333 IC50 = 22000 nM T20251 C1SNE7 62705334 IC50 = 5300 nM T20251 C2O6FQ 62705335 IC50 = 3400 nM T20251 CTM29C 62705504 IC50 = 5700 nM T20251 CZHO61 62705505 IC50 = 7900 nM T20251 CT41VY 62705506 IC50 = 6300 nM T20251 CP9HO0 62705507 IC50 = 4400 nM T20251 CSHR51 62705508 IC50 = 1900 nM T20251 CVPW40 62705509 IC50 = 3400 nM T20251 CA4RU3 62706110 IC50 = 1600 nM T20251 CM0Z3B 62707610 IC50 = 7300 nM T20251 CZDW91 65458453 IC50 > 16000 nM T20251 C9SEG5 65458673 IC50 > 16000 nM T20251 CC82DM 65459349 IC50 = 1800 nM T20251 C0JSU4 65459575 IC50 > 16000 nM T20251 CVUT64 66549717 IC50 = 4080 nM T20251 C1MDS9 66549721 IC50 = 13970 nM T20251 C6EJ3F 66551245 IC50 = 25118.86 nM T20251 CBI4P9 66551368 IC50 = 290 nM T20251 C3SCF6 66551759 IC50 = 870 nM T20251 C2LBW7 66551925 IC50 > 30000 nM T20251 CLHX28 66553128 IC50 = 27000 nM T20251 CA42UL 66554658 IC50 = 15848.93 nM T20251 CX25QN 66555696 IC50 > 50118.72 nM T20251 CL0X8S 66555697 IC50 > 50118.72 nM T20251 C2Y7FX 66555698 IC50 = 25118.86 nM T20251 C8PST7 66556032 IC50 = 10000 nM T20251 CV8JO4 66556033 IC50 > 50118.72 nM T20251 CSZ6I5 66556035 IC50 > 50118.72 nM T20251 C6SL1Q 66556036 IC50 > 50118.72 nM T20251 CX6J3B 66556201 IC50 = 25118.86 nM T20251 CHWG72 66556203 IC50 = 39810.72 nM T20251 CVPT78 66556206 IC50 = 50118.72 nM T20251 C0F5HW 66556207 IC50 > 50118.72 nM T20251 C6E7CU 66556365 IC50 = 12589.25 nM T20251 CR7JT9 66556366 IC50 = 31622.78 nM T20251 CSM89V 66556371 IC50 = 5011.87 nM T20251 CK9QI1 66556533 IC50 = 19952.62 nM T20251 CA1Z4Q 66556534 IC50 > 50118.72 nM T20251 CNRZ13 66556535 IC50 > 50118.72 nM T20251 C7MD5X 66556536 IC50 = 15848.93 nM T20251 CL3EN2 66556938 IC50 > 10000 nM T20251 CUC7B3 66557964 IC50 = 45000 nM T20251 C85RBC 66559553 IC50 = 1900 nM T20251 C95GNE 66559554 IC50 = 2700 nM T20251 CKW13M 66559641 IC50 = 4300 nM T20251 CP1BI4 66559642 IC50 = 30000 nM T20251 C3MW0K 66559643 IC50 = 1100 nM T20251 C0TL3Y 66559644 IC50 > 30000 nM T20251 CXS5D6 66590299 Ki = 9520 nM T20251 CHO3M7 66597981 IC50 > 30000 nM T20251 C7W2XF 66597997 IC50 > 30000 nM T20251 C52HRW 66598095 IC50 > 30000 nM T20251 C1ET4P 66598128 IC50 = 1900 nM T20251 C5D3TJ 66598153 IC50 > 30000 nM T20251 CZF76R 66608383 IC50 > 10000 nM T20251 CECR98 66615606 IC50 = 15848.93 nM T20251 C9IQ1Y 66615619 IC50 > 31622.78 nM T20251 CA59FS 66615678 IC50 > 31622.78 nM T20251 CL69HQ 66615705 IC50 > 31622.78 nM T20251 CLA3R9 66645269 IC50 > 33000 nM T20251 COTD35 66667669 Ki > 30000 nM T20251 CXSA80 66671848 IC50 > 10000 nM T20251 CZKV14 66679405 IC50 = 2000 nM T20251 CJ0KL5 66679507 IC50 > 10000 nM T20251 C9RS5B 66679618 IC50 = 1800 nM T20251 CUC7E1 66679703 IC50 > 10000 nM T20251 C4TQP9 66688557 IC50 = 12200 nM T20251 C3FG4T 66688815 IC50 = 10300 nM T20251 CKR1D0 66693299 IC50 = 24900 nM T20251 C9BF6L 66797369 IC50 = 72000 nM T20251 C78XLS 66813470 IC50 = 10000 nM T20251 CAOB97 66813557 IC50 = 6309.57 nM T20251 C89WUE 66813671 IC50 = 12589.25 nM T20251 CPK67V 66813703 IC50 = 3981.07 nM T20251 C7DX6Z 66813839 IC50 = 6309.57 nM T20251 CH2D5F 66813859 IC50 = 25118.86 nM T20251 C90OSR 66813870 IC50 = 15848.93 nM T20251 COZ0U9 66813914 IC50 = 7943.28 nM T20251 C5OTD2 66813927 IC50 = 10000 nM T20251 C39PEZ 66814019 IC50 = 25118.86 nM T20251 CG80RS 66814110 IC50 = 15848.93 nM T20251 C5BU7L 66829310 IC50 > 30000 nM T20251 CPZQ50 66829372 IC50 = 1900 nM T20251 C38BYQ 66829396 IC50 > 30000 nM T20251 CEVJ65 66829417 IC50 > 30000 nM T20251 CBE2J9 66829485 IC50 = 12000 nM T20251 CRI63W 66829595 IC50 = 12700 nM T20251 CD1BQ8 66829616 IC50 > 30000 nM T20251 C8OZR1 66829709 IC50 > 30000 nM T20251 CEQ7A6 66829716 IC50 = 2560 nM T20251 CMAD65 66829757 IC50 = 10200 nM T20251 C95TOQ 66855889 IC50 = 794 nM T20251 C85HLV 67011331 IC50 > 30000 nM T20251 C1HSE0 67035086 IC50 = 420 nM T20251 CWI6K5 67035106 IC50 = 1100 nM T20251 C38RGB 67035556 IC50 = 3600 nM T20251 CFM6H7 67049587 IC50 > 100000 nM T20251 CJMU80 67055888 IC50 > 80000 nM T20251 C3VFY7 67104025 IC50 = 19000 nM T20251 CV6Z2X 67204288 IC50 > 10000 nM T20251 CD3C7S 67204380 IC50 = 29000 nM T20251 C7CDA0 67220645 IC50 = 20000 nM T20251 C7V8QD 67251061 IC50 = 20 nM T20251 C3WJ5C 67260498 IC50 > 10000 nM T20251 CKQ9W2 67264691 IC50 = 7620 nM T20251 C3F2JN 67264841 IC50 = 2230 nM T20251 C38ROH 67264950 IC50 = 22100 nM T20251 C3CAR6 67265132 IC50 > 30000 nM T20251 C3Q6ZA 67282848 IC50 = 2200 nM T20251 C4R1IH 67283149 IC50 > 10000 nM T20251 C9LI0M 67294297 IC50 > 30000 nM T20251 CBK9T7 67325548 IC50 = 2100 nM T20251 C2NEB3 67339181 IC50 = 10715.19 nM T20251 CKMV48 67345882 IC50 > 100000 nM T20251 CO3ND7 67387844 Ki > 15000 nM T20251 C36MVU 67389741 IC50 = 16000 nM T20251 C4R8OG 67401728 IC50 = 1100 nM T20251 CPV39L 67406727 IC50 = 47000 nM T20251 C7XU0T 67425014 IC50 > 10000 nM T20251 CBFE84 67436561 Ki > 15000 nM T20251 CZC9M5 67469084 IC50 = 7445 nM T20251 CX60UI 67472601 IC50 = 27500 nM T20251 C37YHJ 67496729 IC50 > 30000 nM T20251 CL9JR7 67516635 IC50 = 1300 nM T20251 CIB4Y6 67516958 IC50 = 7100 nM T20251 COH79P 67517411 IC50 = 150 nM T20251 C0WAQ6 67517817 IC50 = 3000 nM T20251 C02TCR 67518221 IC50 = 420 nM T20251 CF3GR9 67538211 IC50 = 26000 nM T20251 CNB15W 67607112 IC50 > 10000 nM T20251 COM54X 67775149 IC50 = 8500 nM T20251 C32GEY 67922794 IC50 > 10000 nM T20251 CY3AZ9 67960061 IC50 = 3700 nM T20251 C3ARI1 67972106 IC50 = 46000 nM T20251 CXJ68U 67972107 IC50 = 55000 nM T20251 CB05ID 67972431 IC50 > 60000 nM T20251 C5K7QG 67974411 IC50 > 10000 nM T20251 CC28AD 68003782 IC50 = 28400 nM T20251 CXU2T6 68003962 IC50 = 16900 nM T20251 C7ZA5Y 68003997 IC50 = 35100 nM T20251 CQ4M8Y 68004002 IC50 > 50000 nM T20251 CB7T0X 68004010 IC50 = 37500 nM T20251 C9SZT4 68004011 IC50 = 28500 nM T20251 C9BFS2 68004012 IC50 > 50000 nM T20251 CX0B4G 68004016 IC50 > 50000 nM T20251 C6U9NR 68004034 IC50 > 50000 nM T20251 C8EM6J 68004094 IC50 = 11200 nM T20251 CCO4A2 68004146 IC50 = 13400 nM T20251 CO6W9D 68004741 IC50 > 10000 nM T20251 CB6U7F 68005465 IC50 > 10000 nM T20251 CK83VI 68005486 IC50 > 10000 nM T20251 C1RJ7Y 68005600 IC50 > 10000 nM T20251 COX3U9 68005621 IC50 = 8600 nM T20251 C57DTK 68045182 IC50 > 30000 nM T20251 CBOF40 68046989 IC50 = 2900 nM T20251 CG24FU 68071359 IC50 = 120 nM T20251 CG2QU1 68071450 IC50 = 9 nM T20251 CNS57A 68071672 IC50 = 2800 nM T20251 CJ8Y2W 68071788 IC50 = 25 nM T20251 CR5BI7 68071790 IC50 = 110 nM T20251 C3DZ1N 68071887 IC50 = 460 nM T20251 CTL92R 68083077 IC50 = 5900 nM T20251 C0PQL8 68094634 IC50 > 100000 nM T20251 CKJ13C 68095253 IC50 = 13000 nM T20251 CW23LG 68154393 IC50 = 49100 nM T20251 C4KYJ9 68171468 IC50 = 4900 nM T20251 C8T4IB 68199725 IC50 = 2200 nM T20251 C73IYJ 68199726 IC50 = 690 nM T20251 CV0P7D 68199727 IC50 = 1200 nM T20251 CY41JC 68199728 IC50 = 1000 nM T20251 C80ARK 68199735 IC50 = 1900 nM T20251 C7NM8D 68199737 IC50 = 8400 nM T20251 CZ3LH9 68199741 IC50 = 180 nM T20251 CUZX17 68204888 IC50 = 4600 nM T20251 C3K4RT 68204896 IC50 = 20000 nM T20251 CWTD61 68204898 IC50 = 6200 nM T20251 C5QZG7 68204899 IC50 = 2700 nM T20251 CF59AG 68204902 IC50 = 3100 nM T20251 CLS7H4 68204905 IC50 = 8400 nM T20251 CM58CG 68204907 IC50 = 6700 nM T20251 CNTP78 68204921 IC50 > 80000 nM T20251 C7V2SY 68204942 IC50 = 4600 nM T20251 C32QIB 68204998 IC50 = 4800 nM T20251 C4SWU5 68205000 IC50 > 80000 nM T20251 CZQ8R4 68205062 IC50 > 80000 nM T20251 CVA87O 68230212 IC50 > 30000 nM T20251 CYR38C 68241014 IC50 = 6600 nM T20251 C0DEM2 68254010 IC50 = 15000 nM T20251 C17JAZ 68284084 IC50 > 30000 nM T20251 CO48FM 68287853 Ki > 9182 nM T20251 C06RFV 68288164 Ki > 15219 nM T20251 CO6Z7D 68288263 Ki > 9182 nM T20251 C4M9LX 68289700 IC50 > 50118.72 nM T20251 C07JAL 68290083 IC50 > 50118.72 nM T20251 CC70KY 68290508 IC50 > 50118.72 nM T20251 CV9Q6N 68305341 IC50 = 10400 nM T20251 C8V0QK 68305342 IC50 > 11000 nM T20251 CIB52Q 68309298 IC50 > 50118.72 nM T20251 CBGL83 68309299 IC50 > 50118.72 nM T20251 CWDS89 68310172 IC50 > 50118.72 nM T20251 CI6YC4 68378925 IC50 > 30000 nM T20251 CI7S6T 68378958 IC50 = 25000 nM T20251 CU71NC 68379030 IC50 = 24000 nM T20251 C7CBD4 68379135 IC50 = 19000 nM T20251 CT32VB 68379165 IC50 = 23000 nM T20251 CBD8C9 68379213 IC50 = 2100 nM T20251 CLBY90 68380304 IC50 = 9200 nM T20251 CA9MK4 68432911 IC50 = 12000 nM T20251 CA7UZ6 68434755 IC50 = 9000 nM T20251 CQ38HU 68437484 IC50 > 30000 nM T20251 CGM78B 68472574 IC50 > 33000 nM T20251 CB8O4N 68475743 IC50 > 33000 nM T20251 C52HIW 68483436 IC50 = 9400 nM T20251 CEL85X 68483794 IC50 = 1800 nM T20251 CWE97U 68490431 IC50 > 100000 nM T20251 CM61LR 68495004 IC50 = 6000 nM T20251 C0OPQ6 68495695 IC50 = 2100 nM T20251 CXS64A 68502671 IC50 > 31600 nM T20251 C4XJ6F 68513796 IC50 > 100000 nM T20251 C3H7AJ 68513937 IC50 = 15000 nM T20251 C5QB6P 68528423 IC50 = 6000 nM T20251 C4B8KQ 68529738 IC50 = 3700 nM T20251 C85NIY 68533570 IC50 = 4600 nM T20251 C7MB8R 68591735 IC50 > 10000 nM T20251 CM5ZS8 68592173 IC50 > 10000 nM T20251 C2J0MD 68592299 IC50 > 10000 nM T20251 C8YG7Z 68592484 IC50 = 6835 nM T20251 C54QNY 68592631 IC50 = 7551 nM T20251 C6UW1R 68592632 IC50 > 10000 nM T20251 CP29IA 68592826 IC50 < 1000 nM T20251 C2GSP7 68593153 IC50 = 10000 nM T20251 C2PJN0 68593295 IC50 > 10000 nM T20251 C62QGB 68593458 IC50 = 10000 nM T20251 C1Q2UZ 68593479 IC50 = 7711 nM T20251 CKQ4O9 68593622 IC50 = 4580 nM T20251 CSQY72 68593732 IC50 > 10000 nM T20251 C2VIM9 68593774 IC50 > 10000 nM T20251 CE6X8W 68593871 IC50 > 10000 nM T20251 C0MYB6 68653619 IC50 > 33000 nM T20251 CH3Z7F 68658979 IC50 = 600 nM T20251 CYV20U 68728631 IC50 = 3700 nM T20251 CD3U6K 68731121 IC50 = 10500 nM T20251 CCB1T5 68764898 IC50 = 1800 nM T20251 C70QJS 68767049 IC50 = 14000 nM T20251 C8XT7M 68767109 IC50 > 80000 nM T20251 CP23JT 68767124 IC50 > 80000 nM T20251 CKWJ72 68767577 IC50 > 80000 nM T20251 C8U1DK 68767802 IC50 > 80000 nM T20251 CRM71Y 68768923 IC50 > 80000 nM T20251 C6L3ZT 68769143 IC50 > 80000 nM T20251 CHS3Z2 68769744 IC50 = 77000 nM T20251 CTL0O6 68770301 IC50 > 33000 nM T20251 CUVF59 68770356 IC50 = 24000 nM T20251 CT2D3M 68772321 IC50 = 32000 nM T20251 CX5Q2G 68772765 IC50 > 33000 nM T20251 CM92FU 68773430 IC50 = 27000 nM T20251 CZ07NC 68773726 IC50 > 33000 nM T20251 C16VTD 68774064 IC50 = 45000 nM T20251 CR28FH 68774353 IC50 > 33000 nM T20251 CWV13E 68774423 IC50 = 30000 nM T20251 C5J1XL 68774942 IC50 > 33000 nM T20251 C59FDP 68775014 IC50 > 31000 nM T20251 C23PDV 68775184 IC50 > 33000 nM T20251 CL6N2D 68775231 IC50 > 33000 nM T20251 CC98XW 68775928 IC50 = 56000 nM T20251 C89CQS 68779277 EC50 > 10000 nM T20251 CG46AF 68816399 IC50 = 1200 nM T20251 C9S1NP 68818964 IC50 = 1100 nM T20251 C6FZD0 68846936 IC50 = 25118.86 nM T20251 CZPM30 68849581 IC50 > 31622.78 nM T20251 C3YW1K 68860750 IC50 > 1000 nM T20251 C1UMP9 68867935 IC50 = 60000 nM T20251 C5PY2V 68938028 IC50 > 25118.86 nM T20251 C8Y3PB 68963393 IC50 = 700 nM T20251 C1KAN5 68963686 IC50 = 1600 nM T20251 C52BVJ 68963698 IC50 > 10000 nM T20251 CWZU52 68988296 IC50 > 80000 nM T20251 CBH6T3 69003776 IC50 = 14000 nM T20251 CG6JX0 69010662 IC50 > 31600 nM T20251 C9SFL1 69011426 IC50 = 2100 nM T20251 CYIB47 69012259 IC50 = 5900 nM T20251 CF57OD 69012280 IC50 = 3800 nM T20251 CI8GH6 69013596 IC50 = 4900 nM T20251 C6IP8Q 69082816 IC50 = 12000 nM T20251 C5CB4U 69087439 IC50 = 33000 nM T20251 CJM2Y1 69087440 IC50 = 10000 nM T20251 CZ0IC8 69087441 IC50 = 60000 nM T20251 C08ZXY 69087444 IC50 = 3400 nM T20251 CAIG78 69087446 IC50 = 3400 nM T20251 C57NKJ 69087450 IC50 = 8500 nM T20251 CX2U1Z 69087451 IC50 = 12000 nM T20251 C04OLI 69087452 IC50 = 52000 nM T20251 C59HRV 69087454 IC50 = 4500 nM T20251 C1O4EV 69087469 IC50 = 9100 nM T20251 CXV98R 69087490 IC50 = 31000 nM T20251 C1XE4Q 69087494 IC50 = 8200 nM T20251 CGQ40U 69087495 IC50 = 13000 nM T20251 CCO97X 69087505 IC50 = 27000 nM T20251 CI3A6W 69087537 IC50 = 100000 nM T20251 CMA21H 69087541 IC50 = 49000 nM T20251 CQF9T5 69087543 IC50 = 68000 nM T20251 CVG42E 69087545 IC50 = 22000 nM T20251 CG31FX 69087546 IC50 = 33000 nM T20251 CX3P0T 69087562 IC50 = 17000 nM T20251 CXF5P9 69213151 IC50 = 7943.28 nM T20251 C07YOG 69260079 IC50 = 31622.78 nM T20251 CV7P3D 69260851 IC50 = 31622.78 nM T20251 C4QO7E 69260946 IC50 = 31622.78 nM T20251 CO9U3M 69262172 IC50 = 1584.89 nM T20251 C7HN5L 69272932 IC50 = 31622.78 nM T20251 CJ2D3I 69274365 IC50 = 31622.78 nM T20251 CPGC67 69285465 IC50 > 80000 nM T20251 CM5XA1 69285531 IC50 = 32000 nM T20251 C0QZ4U 69285563 IC50 > 80000 nM T20251 C5T2GC 69285794 IC50 = 360 nM T20251 C8R4LZ 69286108 IC50 = 5300 nM T20251 CNT95I 69286635 IC50 = 2700 nM T20251 COD5Y1 69347575 IC50 = 15848.93 nM T20251 C51DQR 69347707 IC50 = 31622.78 nM T20251 C8F1CY 69347719 IC50 = 12589.25 nM T20251 C93COF 69347980 IC50 = 19952.62 nM T20251 CPW42A 69348078 IC50 = 25118.86 nM T20251 C6Z7UL 69435853 IC50 = 600 nM T20251 C6XQ3C 69439557 IC50 = 600 nM T20251 CGD48T 69513487 IC50 = 2000 nM T20251 C6RV9Y 69513502 IC50 = 110 nM T20251 C0NAD7 69513622 IC50 = 2000 nM T20251 C25HXG 69513678 IC50 = 5000 nM T20251 COSH07 69513688 IC50 = 100 nM T20251 CKE4H3 69513748 IC50 = 5000 nM T20251 C2AZ4X 69787126 IC50 = 3981.07 nM T20251 CC8QU9 70227534 IC50 > 10000 nM T20251 CI0XF8 70274815 IC50 > 100000 nM T20251 CCG16F 70276365 IC50 = 25118.86 nM T20251 CE1J0O 70276811 IC50 = 15848.93 nM T20251 C06WFN 70276830 IC50 > 100000 nM T20251 CDQ85E 70276990 IC50 > 100000 nM T20251 CGET13 70278898 IC50 = 31622.78 nM T20251 C2GT5H 70280758 IC50 > 100000 nM T20251 CA6DM2 70281073 IC50 > 100000 nM T20251 CK26FY 70295607 IC50 = 4400 nM T20251 CV4X5S 70295927 IC50 > 30000 nM T20251 CXD5V6 70297609 IC50 = 260 nM T20251 C5ZSV0 70355830 Ki = 5220 nM T20251 C7VJ6A 70647728 IC50 = 10000 nM T20251 CC63NT 70675147 IC50 = 37000 nM T20251 CYM94S 70676472 IC50 = 2200 nM T20251 C7J0FD 70676474 IC50 = 980 nM T20251 CLTA38 70676476 IC50 = 830 nM T20251 CMN57J 70676478 IC50 = 180 nM T20251 C9QZ7C 70676480 IC50 = 1560 nM T20251 CN12IT 70680969 IC50 = 2500 nM T20251 C0VEM7 70680970 IC50 = 6500 nM T20251 CP8XS4 70681040 Ki = 1400 nM T20251 CF85AB 70681063 Ki = 2460 nM T20251 C9LW7K 70681064 Ki = 950 nM T20251 CS8V7G 70681068 Ki = 730 nM T20251 CA27SR 70681184 IC50 > 10000 nM T20251 C23CRI 70681196 IC50 = 5350 nM T20251 CEP43U 70681217 IC50 = 1200 nM T20251 C4AX2B 70681647 IC50 = 900 nM T20251 C3MBU1 70681648 IC50 = 10 nM T20251 C71XOI 70681872 IC50 > 100000 nM T20251 C4KWV3 70682467 IC50 = 9800 nM T20251 CSM23I 70682523 IC50 > 10000 nM T20251 CZ84UX 70682584 IC50 > 100000 nM T20251 C8D6ZB 70683088 IC50 = 1600 nM T20251 CKM4C2 70683089 IC50 = 13000 nM T20251 C7BPF4 70683090 IC50 = 3600 nM T20251 CRTD40 70683091 IC50 = 2000 nM T20251 CJV64I 70683156 Ki = 160 nM T20251 C9BR3A 70683161 Ki = 2900 nM T20251 CN79ZX 70683165 Ki = 1900 nM T20251 C94GTH 70683168 Ki = 2800 nM T20251 C3ZY6F 70683178 Ki = 1400 nM T20251 C6QC5J 70683184 Ki = 300 nM T20251 CK6JM8 70683187 Ki = 980 nM T20251 C1UBD3 70683285 IC50 = 21900 nM T20251 C3NR1Z 70683781 IC50 = 300 nM T20251 C1ARO8 70684544 IC50 = 15848.93 nM T20251 C6CWV8 70684549 IC50 = 100 nM T20251 C9F5ZM 70684550 IC50 = 3500 nM T20251 CKN95T 70685174 IC50 = 2900 nM T20251 CUQ92A 70685175 IC50 = 1200 nM T20251 CIV4S6 70685239 Ki = 50 nM T20251 CLW68N 70685259 Ki = 2500 nM T20251 C2IDQ6 70685264 Ki = 1500 nM T20251 CO1ZR5 70685266 Ki = 600 nM T20251 CRP7Z1 70685269 Ki = 2900 nM T20251 CWIC42 70685308 IC50 = 28800 nM T20251 CNH04A 70685394 IC50 = 20800 nM T20251 CG1MS3 70685518 IC50 = 28000 nM T20251 C8HF3M 70685675 IC50 = 93200 nM T20251 C3UO2F 70686000 IC50 = 33000 nM T20251 C0NMH8 70686404 IC50 = 13400 nM T20251 C7OX5Z 70686473 IC50 > 33000 nM T20251 CYO5N3 70686766 IC50 > 25000 nM T20251 CL9RE3 70686820 IC50 > 100000 nM T20251 C65EDY 70686822 IC50 > 100000 nM T20251 CY0N4S 70687331 IC50 = 2600 nM T20251 C84GET 70687332 IC50 = 7000 nM T20251 CI0Z9V 70687389 Ki = 320 nM T20251 CEAK85 70687392 Ki = 800 nM T20251 C3E9VJ 70687415 Ki = 1100 nM T20251 C0A3VH 70687418 Ki = 2300 nM T20251 C0YZF1 70687477 IC50 = 3700 nM T20251 C9V6ML 70687502 Ki = 30000 nM T20251 CL8W4C 70687532 IC50 = 1920 nM T20251 C85ORZ 70687534 IC50 = 200 nM T20251 CFO9M4 70687535 IC50 = 5480 nM T20251 CX58LB 70688042 IC50 = 800 nM T20251 CWO02R 70688127 IC50 = 16300 nM T20251 CIS85H 70688149 IC50 = 5600 nM T20251 C4VU7J 70688210 IC50 > 60000 nM T20251 CR80CD 70688263 IC50 = 2100 nM T20251 CD2EW1 70688785 IC50 > 31622.78 nM T20251 C1GN5V 70688791 IC50 = 120 nM T20251 CA7PZ9 70688792 IC50 = 100 nM T20251 C17MXW 70688793 IC50 = 240 nM T20251 C5IYR0 70688897 IC50 > 100000 nM T20251 CL68HK 70689385 IC50 = 4200 nM T20251 CBY8T6 70689386 IC50 = 2800 nM T20251 CTJL92 70689387 IC50 = 15000 nM T20251 C6YJL1 70689452 Ki = 1100 nM T20251 CO89VX 70689473 Ki = 1200 nM T20251 CM3PD8 70689475 Ki = 2200 nM T20251 CIE2O6 70689591 IC50 = 6270 nM T20251 CHAV16 70689592 IC50 = 40800 nM T20251 CMGO80 70689593 IC50 = 13100 nM T20251 CVYC02 70689594 IC50 = 3300 nM T20251 C9RDP5 70689914 IC50 > 30000 nM T20251 C0QUO1 70689915 IC50 > 30000 nM T20251 CV82BX 70690866 IC50 = 7943.28 nM T20251 CVSJ38 70690870 IC50 = 25 nM T20251 CY6E2Q 70691339 IC50 = 1400 nM T20251 CV2T7S 70691408 IC50 = 1040 nM T20251 CJY73E 70691486 IC50 = 3000 nM T20251 CV8QT4 70691487 IC50 = 2000 nM T20251 C8R0SZ 70691558 Ki = 1100 nM T20251 CRXG05 70691559 Ki = 1200 nM T20251 CYJ3F6 70691560 Ki = 100 nM T20251 CK6I2V 70691577 Ki = 1500 nM T20251 C7ET5J 70691581 Ki = 990 nM T20251 CJ85NC 70691582 Ki = 930 nM T20251 C27IPY 70691584 Ki = 1100 nM T20251 C2N1MW 70691706 IC50 = 430 nM T20251 C14ZJR 70691707 IC50 = 840 nM T20251 C27ECJ 70691721 IC50 = 2500 nM T20251 C0XRC9 70691981 IC50 = 76000 nM T20251 C7ASK8 70692129 IC50 > 32000 nM T20251 C2GXN6 70692344 IC50 = 1600 nM T20251 CZOF81 70693115 IC50 = 6309.57 nM T20251 CMFW03 70693116 IC50 = 25118.86 nM T20251 C5RSJ0 70693117 IC50 = 25118.86 nM T20251 CM4P5Z 70693582 IC50 = 2100 nM T20251 CA9R2G 70693583 IC50 = 4500 nM T20251 C35ASU 70693584 IC50 = 1300 nM T20251 C8JUY5 70693585 IC50 = 7600 nM T20251 CX0E3Y 70693586 IC50 = 4700 nM T20251 CLN9F4 70693648 Ki = 900 nM T20251 CM3LU4 70693649 Ki = 2000 nM T20251 C3GVN0 70693667 IC50 = 760 nM T20251 CKP02Q 70693669 Ki = 1200 nM T20251 C6N3DT 70693670 Ki = 2750 nM T20251 C6GCU1 70693673 Ki = 1800 nM T20251 CHUE45 70693674 Ki = 680 nM T20251 C6P3XM 70693710 IC50 = 2700 nM T20251 CR30DQ 70693785 IC50 = 250 nM T20251 C52LMB 70693791 IC50 = 870 nM T20251 C7HW2B 70694179 IC50 > 33000 nM T20251 C1VS0O 70694288 IC50 = 750 nM T20251 C65FHO 70694723 IC50 > 30000 nM T20251 CCQ49A 70695045 IC50 = 12589.25 nM T20251 C63MTE 70695047 IC50 > 31622.78 nM T20251 C2O7WF 70695089 IC50 = 21500 nM T20251 C75YPE 70695115 IC50 > 25000 nM T20251 C01IDC 70695171 IC50 > 100000 nM T20251 C5T6JA 70695705 IC50 = 10000 nM T20251 CEK60M 70695761 Ki = 430 nM T20251 CX6L3G 70695764 Ki = 500 nM T20251 CF4HZ3 70695774 IC50 = 510 nM T20251 CBHD70 70695780 Ki = 3200 nM T20251 CZL9G2 70695782 Ki = 2300 nM T20251 CUL37Y 70695784 Ki = 2400 nM T20251 C26OHM 70695785 Ki = 1000 nM T20251 CD1V2W 70695786 Ki = 320 nM T20251 CFB1W2 70695912 IC50 = 31900 nM T20251 CB50NG 70696261 IC50 > 33000 nM T20251 C3GDX9 70696694 IC50 > 30000 nM T20251 CMS6J5 70697098 IC50 = 730 nM T20251 C84WJI 70697099 IC50 = 5100 nM T20251 CT1GF8 70697151 IC50 > 25000 nM T20251 C34WHG 70697225 IC50 > 100000 nM T20251 CBDL19 70792359 IC50 > 30000 nM T20251 C7DO1N 70817239 IC50 > 30000 nM T20251 C6L7FH 70817382 IC50 > 30000 nM T20251 CKP4O8 70855957 IC50 = 8600 nM T20251 CLKU89 70856302 IC50 = 7000 nM T20251 CUCQ24 70874317 EC50 > 100000 nM T20251 C1H7VK 70874453 EC50 = 23000 nM T20251 CJF91M 70874544 EC50 = 13200 nM T20251 C9EWB8 70874603 EC50 = 65000 nM T20251 CF1G3K 70874916 EC50 = 34000 nM T20251 C30AJI 70914208 EC50 = 16000 nM T20251 C2TC8W 70914230 EC50 = 71000 nM T20251 CM65DI 70980530 IC50 = 9000 nM T20251 CH7J2X 70982568 IC50 = 1000 nM T20251 C61DAP 70983443 IC50 = 1200 nM T20251 C9ASG6 70984064 IC50 = 3600 nM T20251 C0O7XS 71007248 IC50 = 2800 nM T20251 CHC04W 71008131 IC50 >= 10000 nM T20251 CX3H4C 71009783 IC50 = 1000 nM T20251 C57SJO 71041303 IC50 = 9300 nM T20251 CZ3BM6 71041781 IC50 = 600 nM T20251 C6HRK0 71041789 IC50 = 5400 nM T20251 C4A8FE 71041792 IC50 = 4470 nM T20251 CGXQ60 71041800 IC50 > 10000 nM T20251 C1X8VO 71041841 IC50 = 9100 nM T20251 C3J4SN 71041846 IC50 > 10000 nM T20251 C9WRL7 71041848 IC50 = 1800 nM T20251 C6SH7U 71041850 IC50 = 6000 nM T20251 CK2ML7 71041874 IC50 = 5800 nM T20251 CGWL13 71041904 IC50 = 7200 nM T20251 CV7DL8 71041905 IC50 = 5500 nM T20251 C9RX6A 71041917 IC50 = 8100 nM T20251 C18RLK 71072034 IC50 = 6309.57 nM T20251 C4C0SP 71072040 IC50 = 15848.93 nM T20251 C1YNH6 71072044 IC50 > 10000 nM T20251 CVU3G7 71072050 IC50 > 31622.78 nM T20251 C2M1JY 71072052 IC50 = 5011.87 nM T20251 CE6Y8Z 71072057 IC50 > 10000 nM T20251 C0Z3KN 71072081 IC50 = 6309.57 nM T20251 C3FR6X 71072104 IC50 = 10000 nM T20251 C1BEC9 71072113 IC50 = 6309.57 nM T20251 CNY09L 71072115 IC50 = 12589.25 nM T20251 CFNZ23 71072118 IC50 >= 10000 nM T20251 C6HRB4 71077940 Ki = 40700 nM T20251 C6NKY5 71078482 Ki = 11000 nM T20251 C50WGF 71078515 Ki = 7000 nM T20251 CQUR63 71089192 IC50 = 21000 nM T20251 CFK50V 71110267 Ki = 4500 nM T20251 CS4T0U 71110270 Ki = 4000 nM T20251 C3ORQ5 71110347 Ki = 4900 nM T20251 C3G7QB 71110423 Ki = 12000 nM T20251 CD80YI 71110425 Ki = 20500 nM T20251 CAH09S 71110518 Ki = 25700 nM T20251 CZ29NF 71113911 IC50 > 50118.72 nM T20251 CT1L2V 71113915 IC50 > 50118.72 nM T20251 C1XHA8 71116039 IC50 = 13000 nM T20251 CC43QK 71151588 IC50 = 6200 nM T20251 CYDQ07 71152634 IC50 = 14000 nM T20251 CV0O7K 71152643 IC50 = 8000 nM T20251 C1SQ5Y 71152646 IC50 = 2.13 nM T20251 CL2DQ6 71152655 IC50 = 1000 nM T20251 CHW5A1 71152656 IC50 = 6100 nM T20251 C9GD1Z 71152689 IC50 = 7900 nM T20251 CTK5F6 71152708 IC50 = 2700 nM T20251 CDI7Y0 71152709 IC50 = 8.75 nM T20251 C40QZK 71152713 IC50 = 320 nM T20251 C8QRW6 71152722 IC50 = 3.87 nM T20251 CFZS36 71152743 IC50 = 2000 nM T20251 CQ1Y5R 71152751 IC50 = 12200 nM T20251 CN1O5A 71152755 IC50 = 1.21 nM T20251 CUA70R 71152803 IC50 = 2400 nM T20251 C5MD0V 71152806 IC50 = 900 nM T20251 CDZ6I8 71152809 IC50 = 23900 nM T20251 C95POA 71152813 IC50 = 4000 nM T20251 CDW0Q6 71152814 IC50 = 25400 nM T20251 CIYU58 71152816 IC50 = 3300 nM T20251 C1HYG6 71152822 IC50 = 29100 nM T20251 C6AI9L 71152823 IC50 = 3700 nM T20251 C7R5CM 71152828 IC50 = 200 nM T20251 CQ1R7G 71152842 IC50 = 2.9 nM T20251 CV83IB 71152846 IC50 = 4260 nM T20251 CD2ZN8 71152850 IC50 = 9400 nM T20251 CLK89J 71152851 IC50 = 5300 nM T20251 C2LRT0 71152860 IC50 = 3200 nM T20251 C9B0LK 71152871 IC50 = 0.73 nM T20251 C2AP9L 71152878 IC50 = 9200 nM T20251 C21SCA 71152890 IC50 = 2900 nM T20251 CMG8Y1 71152895 IC50 = 800 nM T20251 CAD57T 71152903 IC50 = 1.19 nM T20251 CGVW14 71152905 IC50 = 3000 nM T20251 C50BQR 71152932 IC50 = 2400 nM T20251 CDKF43 71152934 IC50 = 700 nM T20251 CJZM06 71152971 IC50 = 370 nM T20251 C6W3UY 71152975 IC50 = 700 nM T20251 C05ODL 71152981 IC50 = 3300 nM T20251 CW5KQ7 71152985 IC50 = 8.35 nM T20251 C2G9IR 71153003 IC50 > 60000 nM T20251 C08EJQ 71153009 IC50 = 17300 nM T20251 CC42ES 71153030 IC50 = 8900 nM T20251 CI50XB 71153035 IC50 > 60000 nM T20251 CD4N6B 71153053 IC50 = 3.21 nM T20251 CALF50 71153055 IC50 = 6300 nM T20251 C3HZ6D 71153063 IC50 = 400 nM T20251 C84NTK 71153068 IC50 = 17500 nM T20251 CRES81 71153070 IC50 = 1300 nM T20251 CAV03R 71153095 IC50 = 5800 nM T20251 CSU6Y5 71153098 IC50 = 800 nM T20251 CH52AF 71153108 IC50 = 24400 nM T20251 CGI67Z 71153155 IC50 = 7600 nM T20251 CRJL31 71153157 IC50 = 1000 nM T20251 CPEC13 71153160 IC50 = 11.46 nM T20251 CK27UL 71153161 IC50 = 1.66 nM T20251 C21IBW 71153175 IC50 = 43500 nM T20251 CC9H1B 71181325 IC50 = 1200 nM T20251 CYXF24 71181326 IC50 = 11000 nM T20251 CS4O1D 71181328 IC50 = 8400 nM T20251 CJY8L3 71181338 IC50 = 2800 nM T20251 C5QVR4 71181386 IC50 = 4.83 nM T20251 C3A2MI 71181421 IC50 = 1400 nM T20251 CKO9P6 71181433 IC50 = 1600 nM T20251 CS7O9E 71181495 IC50 = 900 nM T20251 CM25RB 71181508 IC50 = 2700 nM T20251 CB98GE 71181529 IC50 = 1.78 nM T20251 CM1PL3 71181535 IC50 = 700 nM T20251 C0M1WO 71181547 IC50 > 60000 nM T20251 CX5P1U 71181567 IC50 = 1300 nM T20251 C9UP3L 71181628 IC50 = 7000 nM T20251 CY6V8S 71181641 IC50 = 5500 nM T20251 C32UMV 71203748 IC50 = 40000 nM T20251 CBKF84 71222614 IC50 = 3500 nM T20251 C87MGT 71226277 IC50 = 16000 nM T20251 CLIH32 71226367 IC50 = 4300 nM T20251 CRSA04 71226374 IC50 = 25700 nM T20251 C4J8MI 71226400 IC50 = 16000 nM T20251 CE4Y8J 71226521 IC50 = 2400 nM T20251 COU73Y 71226944 IC50 = 4500 nM T20251 C1WP5Y 71226964 IC50 = 13000 nM T20251 C1B9KV 71227161 IC50 = 12000 nM T20251 CI8E6U 71227163 IC50 = 8900 nM T20251 C7Y2LB 71230234 IC50 > 100000 nM T20251 CSB2N6 71235464 IC50 = 5800 nM T20251 C40JOZ 71235465 IC50 = 24000 nM T20251 CH29GF 71258526 IC50 > 30000 nM T20251 CIR30L 71263305 IC50 > 30000 nM T20251 C9AT8D 71263621 IC50 = 1600 nM T20251 C6BE5X 71271461 IC50 > 30000 nM T20251 C1MVL0 71273460 IC50 > 30000 nM T20251 C0GL4U 71276387 IC50 = 11400 nM T20251 CV7ZP5 71276437 IC50 = 4100 nM T20251 C47QTF 71279423 IC50 > 10000 nM T20251 CZR37K 71279507 IC50 > 2000 nM T20251 CU4P3X 71279543 IC50 > 3000 nM T20251 C5L8SW 71279563 IC50 > 1000 nM T20251 CV96FO 71279672 IC50 = 4150 nM T20251 CKJ58I 71279693 IC50 = 293 nM T20251 CZY5P7 71279859 IC50 = 414 nM T20251 CXZG59 71280008 IC50 = 4100 nM T20251 C5TXH9 71280067 IC50 > 3000 nM T20251 CW0FK6 71280128 IC50 > 30000 nM T20251 CGI01S 71280152 IC50 = 1440 nM T20251 C61BWN 71280407 IC50 > 2000 nM T20251 C5CTH0 71280416 IC50 < 300 nM T20251 C63EIL 71280539 IC50 = 429 nM T20251 CUP25C 71280634 IC50 = 6320 nM T20251 CT1NU9 71283192 IC50 = 4000 nM T20251 C8OGT4 71283628 IC50 > 30000 nM T20251 C4AP9F 71288434 IC50 > 10000 nM T20251 CNVG06 71304813 IC50 > 50000 nM T20251 CWY4S0 71304814 IC50 > 50000 nM T20251 C5DXK1 71307955 IC50 = 5000 nM T20251 CR37DA 71419478 IC50 = 31622.78 nM T20251 C3QUF4 71449241 EC50 = 4600 nM T20251 CBQ8P4 71449250 IC50 = 1258.93 nM T20251 CCX2W5 71449253 IC50 = 42 nM T20251 CR4L9T 71449282 IC50 = 10000 nM T20251 CHF08N 71449283 IC50 = 19952.62 nM T20251 CVY54C 71449294 IC50 = 3981.07 nM T20251 C5SML3 71449452 IC50 = 31622.78 nM T20251 CH5X6M 71449584 IC50 = 12589.25 nM T20251 CH5PX8 71449585 IC50 = 10000 nM T20251 CBIT41 71449750 IC50 > 100000 nM T20251 CDP7T0 71449813 IC50 > 10000 nM T20251 C92RIS 71449970 IC50 = 8500 nM T20251 CHU5V7 71449971 IC50 = 1300 nM T20251 CL64JH 71449972 IC50 = 5500 nM T20251 C5YX9S 71450146 IC50 = 300 nM T20251 CS2W0I 71450257 IC50 = 5500 nM T20251 CQ41UR 71450379 IC50 = 19000 nM T20251 CFPK62 71450420 IC50 = 11500 nM T20251 C6DIL5 71450436 IC50 = 8000 nM T20251 CPDJ19 71450468 Ki = 462 nM T20251 CB83YL 71451044 IC50 = 79.43 nM T20251 C0B7ZW 71451051 IC50 = 150 nM T20251 C0L8PR 71451052 IC50 = 3.1 nM T20251 CE98WI 71451053 IC50 = 67 nM T20251 C9BK1J 71451073 IC50 = 1810 nM T20251 CIFE14 71451076 IC50 = 12589.25 nM T20251 CLSQ82 71451077 IC50 = 31622.78 nM T20251 C0RL3C 71451078 IC50 = 6309.57 nM T20251 CGJ7K0 71451084 IC50 = 19952.62 nM T20251 CI0B8V 71451085 IC50 > 31622.78 nM T20251 C3FC1H 71451390 IC50 > 100000 nM T20251 C4W6YG 71451391 IC50 > 100000 nM T20251 CI1OL6 71451639 IC50 > 100000 nM T20251 CL7P2A 71451832 IC50 = 19000 nM T20251 CZ7R2Y 71451924 Ki = 950 nM T20251 C9AO0Q 71452203 IC50 = 16000 nM T20251 C03DBO 71452204 IC50 = 5000 nM T20251 CW6C9V 71452241 IC50 = 7000 nM T20251 CL01IH 71452297 Ki = 2206 nM T20251 C5ZKN6 71452298 Ki = 44 nM T20251 CHQ1F0 71452299 Ki = 377 nM T20251 CHEB80 71452520 IC50 = 6300 nM T20251 C0YXD3 71452871 IC50 = 1258.93 nM T20251 CY7NM9 71452872 IC50 = 2511.89 nM T20251 C42GQM 71452880 IC50 = 47 nM T20251 C3JZH1 71452881 IC50 = 280 nM T20251 CKMZ80 71452882 IC50 = 4700 nM T20251 CXT57R 71452899 IC50 = 6309.57 nM T20251 COQ0P1 71453071 IC50 = 31622.78 nM T20251 C8C9JT 71453204 IC50 > 100000 nM T20251 C45PHI 71453617 IC50 = 3100 nM T20251 CP74WT 71453805 IC50 > 33000 nM T20251 CT23NI 71453897 IC50 = 22 nM T20251 C3ZLD5 71453913 IC50 = 19700 nM T20251 CC7PH1 71453987 IC50 = 5100 nM T20251 CB43OI 71454008 IC50 = 24000 nM T20251 CZI84F 71454093 Ki = 1638 nM T20251 CLDP69 71454277 IC50 = 11000 nM T20251 C47GYB 71454279 IC50 > 25000 nM T20251 C02FKR 71454296 IC50 = 12589.25 nM T20251 C4JN5I 71454639 IC50 = 3.981 nM T20251 C8Q0JV 71454645 IC50 = 7 nM T20251 C5WU8L 71454670 IC50 = 3981.07 nM T20251 C7XQZ4 71454678 IC50 = 19952.62 nM T20251 CZ4HI3 71455166 IC50 = 7400 nM T20251 C0YD9K 71455398 IC50 = 15000 nM T20251 C8OD4R 71455430 Ki > 10000 nM T20251 C6LH8Q 71455522 IC50 = 1100 nM T20251 CL9YX8 71455523 IC50 = 1800 nM T20251 C8J0WA 71455643 IC50 = 16300 nM T20251 CS2V3E 71455663 IC50 = 8200 nM T20251 CZT0H5 71455744 IC50 = 9500 nM T20251 C8BRU5 71455750 IC50 = 8000 nM T20251 CB0RN5 71455780 IC50 = 13100 nM T20251 C6VDY5 71456055 IC50 = 8300 nM T20251 CMBU21 71456359 IC50 = 251.19 nM T20251 CVT39B 71456360 IC50 = 5011.87 nM T20251 CK87DI 71456361 IC50 = 1258.93 nM T20251 CT7EN2 71456366 IC50 = 22 nM T20251 C3YOV7 71456368 IC50 = 560 nM T20251 C1X6TY 71456401 IC50 = 6309.57 nM T20251 C7AL1C 71456402 IC50 > 25118.86 nM T20251 CORH12 71456403 IC50 = 19952.62 nM T20251 CC3Q9J 71456413 IC50 = 12589.25 nM T20251 CL9BS3 71456722 IC50 > 100000 nM T20251 CT0OQ6 71456725 IC50 = 31622.78 nM T20251 CE2M1B 71456899 IC50 = 23442.29 nM T20251 C6QVT0 71456917 IC50 > 33113.11 nM T20251 C3M9KC 71456918 IC50 > 33113.11 nM T20251 CCF78E 71456919 IC50 = 24547.09 nM T20251 CLO4B6 71456969 IC50 > 100000 nM T20251 CMB6O8 71457147 IC50 = 2900 nM T20251 C7MNB5 71457264 Ki = 800 nM T20251 CQB9F3 71457442 IC50 = 20200 nM T20251 C6PX9L 71457622 Ki = 2189 nM T20251 C1NH9X 71457850 IC50 > 10000 nM T20251 C1EA6Q 71458069 Ki = 18 nM T20251 C3VMS0 71458203 IC50 = 2511.89 nM T20251 C8T5EJ 71458204 IC50 = 158.49 nM T20251 CZ6BX7 71458205 IC50 = 63.1 nM T20251 CI7B2J 71458215 IC50 = 3.9 nM T20251 CK6S7X 71458227 IC50 = 1200 nM T20251 CPST04 71458774 IC50 > 33113.11 nM T20251 CZW7X0 71458868 IC50 > 19952.62 nM T20251 CJ98EQ 71459165 IC50 > 33000 nM T20251 CYL5C6 71459166 IC50 > 33000 nM T20251 C58BIQ 71459167 IC50 = 26800 nM T20251 CV4ZI2 71459168 IC50 = 17500 nM T20251 CY8G0F 71459407 IC50 = 2500 nM T20251 C1LIN4 71459486 IC50 = 1000 nM T20251 COJ85G 71459516 Ki = 2616 nM T20251 CJ1M6I 71459762 IC50 = 2511.89 nM T20251 C89YUI 71460069 IC50 = 150 nM T20251 CYBR37 71460098 IC50 = 7943.28 nM T20251 CQW3L4 71460099 IC50 = 6309.57 nM T20251 CSB76D 71460108 IC50 = 19952.62 nM T20251 CP26GF 71460416 IC50 = 10000 nM T20251 CH51UB 71460419 IC50 = 3981.07 nM T20251 C9LYM0 71460575 IC50 = 19000 nM T20251 CZH53R 71460636 IC50 > 10000 nM T20251 CR2C6Z 71461172 IC50 = 16000 nM T20251 CU9X6E 71461217 IC50 = 30000 nM T20251 C5UB8I 71461218 IC50 = 6000 nM T20251 CETP14 71461260 Ki = 1403 nM T20251 CBSY93 71461487 IC50 > 10000 nM T20251 CEBC62 71461781 IC50 = 15.85 nM T20251 C9DJ1V 71461782 IC50 = 50.12 nM T20251 CV6QH8 71461787 IC50 = 19 nM T20251 CC92TB 71461788 IC50 = 23 nM T20251 CV7ML5 71461830 IC50 = 19952.62 nM T20251 C9UG2X 71462100 IC50 > 100000 nM T20251 CL4MZ5 71462103 IC50 = 10000 nM T20251 CKYO86 71462283 IC50 > 31622.78 nM T20251 CX97KJ 71462389 IC50 > 10000 nM T20251 CZQ4T0 71462891 IC50 = 16400 nM T20251 COT2V4 71462903 IC50 > 33000 nM T20251 C6HN7D 71462955 IC50 = 1000 nM T20251 CG2KF6 71462956 IC50 = 12000 nM T20251 CH2CE8 71462982 Ki = 385 nM T20251 C9R4EX 71462983 Ki = 543 nM T20251 CQ4WG2 71462984 Ki = 300 nM T20251 C7UVZ5 71463198 IC50 = 9500 nM T20251 C0GBL7 71466345 IC50 = 2000 nM T20251 C3YA7I 71466474 IC50 = 47800 nM T20251 C2PMJ7 71474167 Ki = 530 nM T20251 COI42Y 71478198 Ki = 3000 nM T20251 C7MCJ0 71487141 IC50 = 500 nM T20251 CL3S8Q 71487418 IC50 = 11300 nM T20251 CFA9V1 71494937 IC50 = 16000 nM T20251 CCR8J9 71496459 IC50 > 33000 nM T20251 C8V4GQ 71496460 IC50 = 17500 nM T20251 CD64WC 71500036 IC50 > 33000 nM T20251 C1PC8B 71516677 IC50 = 2000 nM T20251 C24ZPL 71516877 IC50 = 5900 nM T20251 CY83FI 71516959 IC50 = 5000 nM T20251 C1N2HF 71517046 IC50 = 1600 nM T20251 C7GS4P 71517047 IC50 = 13000 nM T20251 CWLO57 71517048 IC50 = 5300 nM T20251 C87CZW 71517049 IC50 > 33000 nM T20251 CY0VJ8 71517192 IC50 = 5800 nM T20251 C5S0XY 71517194 IC50 = 6600 nM T20251 C31DLT 71517195 IC50 = 4100 nM T20251 CRG0P7 71517196 IC50 > 33000 nM T20251 CA07TC 71517197 IC50 > 33000 nM T20251 CLAF67 71517240 IC50 > 50000 nM T20251 CYSI71 71517241 IC50 > 50000 nM T20251 C8SR2Q 71517242 IC50 > 50000 nM T20251 C4TGH7 71517401 IC50 > 50000 nM T20251 CU28ZL 71517402 IC50 > 50000 nM T20251 C0BWE4 71517403 IC50 > 50000 nM T20251 CU2TR7 71517573 IC50 > 50000 nM T20251 C1XWC3 71517574 IC50 > 50000 nM T20251 CZ5QD8 71517575 IC50 > 50000 nM T20251 CGE96J 71517576 IC50 > 50000 nM T20251 CFZ27L 71517577 IC50 > 50000 nM T20251 CK81FA 71517737 IC50 > 50000 nM T20251 CVN31I 71518405 IC50 > 50000 nM T20251 CTL9E5 71518406 IC50 = 33500 nM T20251 C9V5RD 71518407 IC50 = 33600 nM T20251 CW39SU 71518408 IC50 = 14700 nM T20251 CH5UM0 71518570 IC50 = 23100 nM T20251 C6DIG9 71518571 IC50 > 50000 nM T20251 CZ0S5X 71518572 IC50 = 47000 nM T20251 CEJ1O6 71518573 IC50 > 50000 nM T20251 CQC14H 71518574 IC50 > 50000 nM T20251 CXV79I 71518727 IC50 = 38900 nM T20251 CMKZ52 71518728 IC50 = 40900 nM T20251 CL05CZ 71518896 IC50 > 50000 nM T20251 C4UMA0 71518897 IC50 = 33300 nM T20251 C3Y2CP 71518898 IC50 = 48900 nM T20251 CGO9T8 71519050 IC50 > 50000 nM T20251 CSU8J9 71519051 IC50 = 46600 nM T20251 C0E9LJ 71519052 IC50 = 46900 nM T20251 CK1GR7 71519053 IC50 = 23500 nM T20251 CGY45E 71519054 IC50 = 42400 nM T20251 C29BZD 71519055 IC50 = 20300 nM T20251 CR1IO9 71519224 IC50 = 27600 nM T20251 CQ8F3O 71519225 IC50 = 33700 nM T20251 CE07SH 71519226 IC50 = 7400 nM T20251 C2FE7Q 71519227 IC50 > 50000 nM T20251 CP25YK 71519381 IC50 > 50000 nM T20251 CZ03XO 71519496 IC50 > 33000 nM T20251 CLQ31I 71519674 Ki > 100000 nM T20251 CLE21W 71520368 IC50 > 33000 nM T20251 C5S0FT 71520369 IC50 > 33000 nM T20251 CZY20B 71520370 IC50 > 33000 nM T20251 C0T9BG 71520371 IC50 > 33000 nM T20251 C3AKL4 71520372 IC50 > 33000 nM T20251 C4OBM9 71520373 IC50 > 33000 nM T20251 CXT3L0 71520486 IC50 > 33000 nM T20251 CA3B5V 71520487 IC50 > 33000 nM T20251 C1HI9J 71520488 IC50 > 33000 nM T20251 C92QDP 71520489 IC50 > 33000 nM T20251 CM6DZ1 71520490 IC50 > 33000 nM T20251 CD1XT8 71520491 IC50 > 33000 nM T20251 CSQH86 71520575 IC50 > 33000 nM T20251 CM1B0W 71523649 IC50 = 14000 nM T20251 C8JC6A 71525586 Ki = 26915.35 nM T20251 CR9ZE5 71525587 Ki > 100000 nM T20251 CRL42M 71525588 Ki = 12882.5 nM T20251 CRM9Q1 71525678 Ki = 34673.69 nM T20251 C2GK7O 71525679 Ki = 43651.58 nM T20251 C7HR1A 71525680 Ki > 100000 nM T20251 C8A0NC 71525681 Ki > 100000 nM T20251 CKU02X 71527981 IC50 = 800 nM T20251 CG7HA3 71528087 IC50 = 3500 nM T20251 CCVD76 71528088 IC50 = 3900 nM T20251 C3O6EK 71529541 IC50 = 17500 nM T20251 C3CT1R 71530223 IC50 > 50000 nM T20251 CE82HN 71533671 IC50 = 3630 nM T20251 CI71DK 71533675 IC50 = 1600 nM T20251 CN8CM1 71533722 IC50 = 24000 nM T20251 C67ZSQ 71540073 IC50 = 4600 nM T20251 CVG8M5 71540729 IC50 = 4700 nM T20251 CWE32H 71540731 IC50 = 20000 nM T20251 C90TFO 71540846 IC50 = 7700 nM T20251 CK2EY7 71540967 IC50 > 33000 nM T20251 C3WR0T 71541076 IC50 > 33000 nM T20251 C0SKF2 71541077 IC50 = 29000 nM T20251 C45CNE 71541078 IC50 = 13000 nM T20251 C3UR6G 71541079 IC50 > 33000 nM T20251 CQ0D2T 71541080 IC50 > 33000 nM T20251 C9VF1X 71541081 IC50 > 33000 nM T20251 CBN7X9 71541082 IC50 > 33000 nM T20251 CJ89BQ 71541083 IC50 = 7800 nM T20251 C9T1HK 71541084 IC50 = 3600 nM T20251 CO26TC 71541094 IC50 = 10000 nM T20251 CE8YO0 71541095 IC50 = 6100 nM T20251 CN79ZY 71541096 IC50 = 10000 nM T20251 CNCR14 71541097 IC50 = 5300 nM T20251 CW34SU 71541098 IC50 = 7600 nM T20251 CKW24J 71541099 IC50 = 10000 nM T20251 C4PYZ6 71541174 IC50 = 6800 nM T20251 C1RZ5T 71541175 IC50 = 3300 nM T20251 CF1B8U 71541176 IC50 = 6600 nM T20251 CU5E7L 71541177 IC50 = 12000 nM T20251 C9I1QA 71541178 IC50 > 33000 nM T20251 CA5O1N 71541179 IC50 = 13000 nM T20251 CZUV57 71541180 IC50 = 21000 nM T20251 C92PZK 71541187 IC50 = 26000 nM T20251 C0T4RD 71541188 IC50 = 15000 nM T20251 CB91FO 71541189 IC50 = 11000 nM T20251 CY5E0J 71541190 IC50 = 21000 nM T20251 C4XK1S 71541191 IC50 = 13700 nM T20251 C32HNI 71541192 IC50 = 15400 nM T20251 C9C0JU 71541193 IC50 > 27000 nM T20251 CFO05K 71541194 IC50 = 26000 nM T20251 CD1T5J 71541195 IC50 = 23000 nM T20251 CXS47M 71541275 IC50 > 33000 nM T20251 C3AFY4 71541276 IC50 > 33000 nM T20251 C98TJN 71541277 IC50 = 15000 nM T20251 C4AG9L 71541278 IC50 > 33000 nM T20251 CVX93I 71541279 IC50 > 33000 nM T20251 C1J4KM 71541280 IC50 > 33000 nM T20251 CBWZ86 71541287 IC50 > 31000 nM T20251 CK82YE 71541288 IC50 > 33000 nM T20251 CQ81HF 71541289 IC50 = 19000 nM T20251 CU53JE 71541292 IC50 > 33000 nM T20251 CR7E4G 71541370 IC50 = 23000 nM T20251 C9IE3U 71541371 IC50 = 13000 nM T20251 CFO83N 71541372 IC50 = 25000 nM T20251 CI6J5K 71541373 IC50 = 12000 nM T20251 CC7YB2 71541376 IC50 = 29000 nM T20251 CWT0Y3 71541468 IC50 = 26000 nM T20251 CGJ86B 71541469 IC50 = 12000 nM T20251 C0CBT4 71541470 IC50 = 13000 nM T20251 CQ8JN9 71541471 IC50 = 18000 nM T20251 CZV7N9 71541472 IC50 = 34000 nM T20251 CL20CV 71541473 IC50 = 9000 nM T20251 C6J9NY 71541572 IC50 = 4300 nM T20251 CS0J6B 71541573 IC50 = 12000 nM T20251 C5CO8Z 71541574 IC50 = 17000 nM T20251 CI90PK 71541575 IC50 = 17000 nM T20251 C4FS8Z 71541576 IC50 = 3100 nM T20251 CSI37G 71541577 IC50 = 9200 nM T20251 C5D6IE 71541687 IC50 = 9000 nM T20251 C3RQP5 71542927 IC50 > 50000 nM T20251 C9N7YA 71544706 IC50 > 32000 nM T20251 C92NEY 71544707 IC50 > 32000 nM T20251 C83YJF 71544946 IC50 > 13000 nM T20251 C2PC6S 71547342 IC50 = 29000 nM T20251 CD97ZU 71547584 IC50 = 1700 nM T20251 CIRZ76 71547586 IC50 = 600 nM T20251 C7V9SQ 71547699 IC50 = 48000 nM T20251 CC0B1F 71547911 IC50 = 6500 nM T20251 CEV53L 71548006 IC50 > 30000 nM T20251 CI7Q4K 71548718 IC50 > 30000 nM T20251 CED62L 71548719 IC50 = 11000 nM T20251 CKB12X 71549359 IC50 = 27000 nM T20251 C4LZM6 71549637 IC50 = 17000 nM T20251 C6JOB5 71549767 IC50 = 5100 nM T20251 CV47CJ 71549769 IC50 = 8000 nM T20251 C5IV9D 71549913 IC50 = 7300 nM T20251 CSHT69 71550657 IC50 > 6000 nM T20251 C7XGD2 71552097 IC50 = 46000 nM T20251 CQ31YB 71552260 IC50 = 32700 nM T20251 CO3WL9 71552261 IC50 = 36100 nM T20251 CHO7D1 71555244 IC50 > 20000 nM T20251 CM04ZX 71555465 IC50 > 20000 nM T20251 C5HK2E 71555534 IC50 > 20000 nM T20251 COW5E6 71560030 IC50 = 13000 nM T20251 CKP12Z 71560031 IC50 = 17400 nM T20251 C6XBY4 71560280 IC50 = 49500 nM T20251 C0FQS4 71560281 IC50 = 2370 nM T20251 C0C5GA 71560284 IC50 > 32000 nM T20251 CYC2W1 71560403 IC50 = 213320 nM T20251 C1WA7E 71560526 IC50 = 21000 nM T20251 C6TEO9 71562957 IC50 = 65300 nM T20251 C0NFT4 71563078 IC50 = 22700 nM T20251 CY74BK 71570778 IC50 = 3950 nM T20251 C6WFT5 71570924 IC50 = 9200 nM T20251 C6SU2O 71572050 Ki = 37700 nM T20251 C14BCP 71572051 Ki = 23400 nM T20251 CB1YS4 71572385 Ki > 60000 nM T20251 CR0KX9 71572386 Ki = 2700 nM T20251 CN52ZY 71572387 Ki = 8600 nM T20251 C2L8XG 71572646 IC50 = 28000 nM T20251 CB2F3M 71573174 IC50 = 7400 nM T20251 C3R0FO 71575419 IC50 > 30000 nM T20251 CUJT21 71582799 IC50 > 100000 nM T20251 CHEZ52 71583033 IC50 = 6600 nM T20251 CNUV80 71583035 IC50 > 25000 nM T20251 CD0K5I 71583037 IC50 > 25000 nM T20251 CQV96E 71583048 IC50 > 33300 nM T20251 CSPR52 71583049 IC50 > 33300 nM T20251 CNT5F3 71583050 IC50 > 33300 nM T20251 CH7I0W 71583051 IC50 > 100000 nM T20251 CAQR82 71583149 IC50 > 25000 nM T20251 CQ16UM 71584055 IC50 > 33000 nM T20251 CWD2Z5 71585566 IC50 > 10000 nM T20251 CNY52I 71586326 Ki = 2000 nM T20251 C5YL7V 71590612 IC50 >= 10000 nM T20251 CH5LE3 71598532 IC50 = 6309.57 nM T20251 CYW46V 71601091 IC50 = 18350 nM T20251 CZS74H 71601235 IC50 > 40000 nM T20251 CAC2V3 71601378 IC50 > 40000 nM T20251 C3XKL2 71603135 Ki = 3388.44 nM T20251 CQ3Y9W 71603136 Ki = 831.76 nM T20251 CA4GQ7 71603139 Ki = 4677.35 nM T20251 CK4T5Q 71603140 Ki = 3630.78 nM T20251 C70OBY 71603141 Ki = 1513.56 nM T20251 C1HEY4 71603142 Ki = 2454.71 nM T20251 CUW27Q 71603194 Ki = 2754.23 nM T20251 C3YA4C 71603551 IC50 = 14800 nM T20251 C6MZO8 71603797 IC50 > 10000 nM T20251 CKY82R 71603916 IC50 = 25200 nM T20251 C9J0EH 71603917 IC50 = 20300 nM T20251 CT8ZS9 71603918 IC50 = 19900 nM T20251 C2X3AO 71603919 IC50 = 12500 nM T20251 CFTR25 71603920 IC50 = 10000 nM T20251 C7BD6V 71603987 IC50 = 75900 nM T20251 C98YDN 71603990 IC50 > 10000 nM T20251 CQ37SD 71604125 IC50 = 59400 nM T20251 CYLF28 71604550 IC50 = 371 nM T20251 CLQ64Y 71604552 IC50 = 208 nM T20251 C5V7WR 71604554 IC50 = 158 nM T20251 CV02ZN 71604556 Ki = 6 nM T20251 C80SAZ 71604558 IC50 = 60 nM T20251 CU6Y8R 71604699 IC50 = 74 nM T20251 CN1EC9 71604700 Ki = 3.5 nM T20251 C8BEX7 71604701 IC50 = 15 nM T20251 CC8PG6 71604703 IC50 > 10 nM T20251 CJ04ZL 71605375 IC50 = 40 nM T20251 C28ZRB 71605376 IC50 > 10000 nM T20251 CJTH01 71605377 IC50 = 146 nM T20251 C7J1QI 71605382 IC50 = 2908 nM T20251 CMZ9J1 71605546 IC50 > 10 nM T20251 CY4MR9 71605549 IC50 = 346 nM T20251 CL9E4D 71605712 IC50 = 53 nM T20251 CT0K3J 71605714 IC50 = 767 nM T20251 C1VE9A 71605716 IC50 = 107 nM T20251 C7L8SH 71605718 IC50 = 135 nM T20251 C08BKQ 71605894 IC50 = 24 nM T20251 CTX0A3 71605896 Ki > 100000 nM T20251 CD3A6U 71606227 IC50 = 285 nM T20251 CZ9AQ8 71606230 Ki = 1208 nM T20251 C4BP5U 71606232 Ki = 86 nM T20251 CB37JD 71606234 IC50 = 377 nM T20251 CW8YG2 71606394 IC50 = 1159 nM T20251 CLBT68 71606396 IC50 = 4019 nM T20251 CZJ74L 71606398 IC50 = 3901 nM T20251 CXM6Z7 71606400 IC50 > 10000 nM T20251 CZ2DN9 71606402 IC50 = 14426 nM T20251 C6WGD4 71606558 IC50 = 14014 nM T20251 CY7S8Z 71606562 Ki = 2460 nM T20251 CX1Z4A 71606712 IC50 = 1992 nM T20251 CJT3H7 71606718 IC50 = 9.9 nM T20251 CI6C2A 71606877 IC50 = 24 nM T20251 C2N0PZ 71606880 IC50 = 86 nM T20251 CBI53Y 71613516 IC50 > 30000 nM T20251 C1Z6JV 71613522 IC50 = 47600 nM T20251 CVBQ58 71614504 IC50 = 30900 nM T20251 CRD4I9 71625797 IC50 = 5400 nM T20251 C5IKR3 71625970 IC50 = 1000 nM T20251 CC54ZM 71625972 IC50 = 6309.57 nM T20251 C5NA4Y 71625975 IC50 = 3981.07 nM T20251 CW7DI6 71626041 IC50 = 1995.26 nM T20251 CGR3I5 71626043 IC50 = 15848.93 nM T20251 CCQ69B 71626102 IC50 = 7943.28 nM T20251 C2WJX0 71626755 IC50 = 10000 nM T20251 CTRE28 71626822 IC50 = 7943.28 nM T20251 C8TID3 71626894 IC50 = 3981.07 nM T20251 C26TXG 71626895 IC50 = 15848.93 nM T20251 C4DHC9 71626896 IC50 = 19952.62 nM T20251 CJV92N 71626898 IC50 = 3981.07 nM T20251 C3XV8I 71626968 IC50 = 5011.87 nM T20251 C7GZI2 71626969 IC50 = 1258.93 nM T20251 CX0VE7 71626971 IC50 = 7943.28 nM T20251 C46RFP 71655299 IC50 > 17500 nM T20251 CDL35U 71655748 IC50 > 10000 nM T20251 CI0GU8 71660496 IC50 = 10900 nM T20251 CA0N8I 71665696 IC50 = 8100 nM T20251 CGD2R7 71680685 IC50 = 7600 nM T20251 CT5L2D 71680688 IC50 = 1500 nM T20251 C6EDG5 71680844 IC50 = 8600 nM T20251 C4C9OW 71680849 IC50 = 9200 nM T20251 C26UGV 71681009 IC50 = 10000 nM T20251 CG2F5B 71681010 IC50 = 12000 nM T20251 CN7ZH6 71681015 IC50 > 33000 nM T20251 C50DHN 71681166 IC50 = 23000 nM T20251 C79QKU 71681209 IC50 = 195 nM T20251 C10OCG 71681315 IC50 = 5700 nM T20251 CRQ1Y6 71681316 IC50 = 2800 nM T20251 C4OU0Y 71681318 IC50 = 1500 nM T20251 C13RPX 71681468 IC50 = 9000 nM T20251 C86XQA 71681473 IC50 = 6150 nM T20251 CU23DO 71681634 IC50 > 33000 nM T20251 C8H2PC 71681635 IC50 = 11000 nM T20251 CH4R7G 71682752 IC50 = 1600 nM T20251 CBVC07 71682893 IC50 = 6000 nM T20251 CFE3Y7 71683044 IC50 = 8000 nM T20251 C3ISR6 71683048 IC50 = 9000 nM T20251 C8LE5D 71695973 IC50 = 22000 nM T20251 CS62NH 71698376 IC50 = 24200 nM T20251 CI8X1R 71698379 IC50 = 12500 nM T20251 CHGS40 71710904 IC50 = 3990 nM T20251 CF6JR1 71711842 IC50 > 3700 nM T20251 CVMG84 71711917 IC50 = 20200 nM T20251 CD3OY7 71711988 IC50 > 33000 nM T20251 C24DMC 71711989 IC50 = 3700 nM T20251 C4L1VN 71713035 IC50 = 14000 nM T20251 C8I9BS 71713478 IC50 = 3700 nM T20251 C9I3GO 71714121 IC50 = 16000 nM T20251 CW7TD2 71716405 IC50 = 2070 nM T20251 COBD81 71716733 IC50 > 33000 nM T20251 C5GE1T 71716742 IC50 > 50000 nM T20251 CWB3V1 71718136 IC50 > 20000 nM T20251 C0O4ID 71718185 IC50 > 33000 nM T20251 CUWM58 71719137 IC50 = 1300 nM T20251 C6YQ4H 71719475 IC50 = 2400 nM T20251 C02FQE 71719561 IC50 > 100000 nM T20251 CG30CF 71719764 IC50 > 50000 nM T20251 C2EWG5 71719830 IC50 > 33000 nM T20251 C1FYA8 71720426 IC50 = 17000 nM T20251 C8IBF0 71720519 IC50 = 5.1 nM T20251 CMI1V5 71720664 IC50 = 7200 nM T20251 CO7B8C 71720776 IC50 = 13000 nM T20251 C30NBJ 71722055 IC50 > 30000 nM T20251 CIN10C 71727133 IC50 = 14500 nM T20251 C73WPT 71730102 Ki = 11890 nM T20251 C7Z1IR 71730238 Ki = 8140 nM T20251 CF78GV 71730361 Ki = 1360 nM T20251 CFHK37 71730881 Ki = 616 nM T20251 CNH38L 71731010 Ki = 1427 nM T20251 CPB1F0 71731512 Ki = 2250 nM T20251 CQ82DI 71731513 Ki > 60000 nM T20251 C60BIX 71763463 IC50 > 100000 nM T20251 CC80KL 71768688 IC50 > 50000 nM T20251 C4KUV6 71768721 IC50 = 43000 nM T20251 C7ZY1J 71768865 IC50 = 5800 nM T20251 CV53CZ 71768899 IC50 > 50000 nM T20251 CKU6V5 71768931 IC50 = 29000 nM T20251 CTSK68 71811225 IC50 > 10000 nM T20251 CVL54T 71811261 IC50 = 4700 nM T20251 COVS02 71812189 IC50 = 1600 nM T20251 C2QT3H 71812413 IC50 = 4000 nM T20251 CZPJ89 71812414 IC50 > 30000 nM T20251 CU1KS7 71812606 IC50 = 17000 nM T20251 CRAB14 71812607 IC50 = 6000 nM T20251 C5JV1P 71812623 IC50 > 100000 nM T20251 CQD1F2 71812796 IC50 = 21000 nM T20251 C2UOA5 71812797 IC50 = 23000 nM T20251 C9NK1C 71812798 IC50 > 30000 nM T20251 C3RE7M 71812799 IC50 = 16000 nM T20251 CD28XR 71816087 IC50 = 9670 nM T20251 CW20HQ 71818431 IC50 > 50000 nM T20251 C2L7TX 71818575 IC50 > 50000 nM T20251 CZ47NP 71819426 IC50 > 33000 nM T20251 C8S3ON 72163808 IC50 > 33000 nM T20251 CPA03W 72163810 IC50 > 33000 nM T20251 CR4B7C 72163925 IC50 = 19000 nM T20251 CQFI71 72163926 IC50 = 16000 nM T20251 CU64GF 72163928 IC50 > 33000 nM T20251 CYNV72 72163929 IC50 = 19000 nM T20251 CK0TQ3 72163930 IC50 = 11000 nM T20251 CCHA62 72164043 IC50 = 16000 nM T20251 CG4M7N 72164287 IC50 > 33000 nM T20251 CZ7YO2 72164288 IC50 > 33000 nM T20251 CDKV52 72164289 IC50 > 33000 nM T20251 CJP4N6 72164290 IC50 > 33000 nM T20251 CE19XB 72164409 Ki = 3520 nM T20251 CB2NP7 72165228 IC50 = 26000 nM T20251 CH68XV 72188554 IC50 > 30000 nM T20251 CO15AV 72188905 IC50 > 30000 nM T20251 C1ERA6 72192163 IC50 = 5000 nM T20251 CD85OH 72201590 IC50 = 1100 nM T20251 C5KTR3 72201875 IC50 = 9 nM T20251 C1N7LQ 72202249 IC50 > 30000 nM T20251 CKMZ39 72202597 IC50 = 5000 nM T20251 CO5XJ3 72202738 IC50 = 3700 nM T20251 C9XL7F 72202747 IC50 > 10000 nM T20251 CJTS50 72202874 IC50 = 8100 nM T20251 CXLR81 72203284 IC50 > 30000 nM T20251 CA10KU 72205492 IC50 = 10230 nM T20251 C78TDP 72205494 IC50 = 9560 nM T20251 CB19LS 72205495 IC50 = 11490 nM T20251 C2PBS7 72375648 IC50 = 46 nM T20251 C23VDP 72375650 IC50 = 32000 nM T20251 CRZ48N 72375747 IC50 = 2500 nM T20251 C6W8VM 72375748 IC50 = 6500 nM T20251 CU9DR1 72375749 IC50 = 27000 nM T20251 CA0Y6E 72375832 IC50 = 5100 nM T20251 CKS9M4 72375834 IC50 = 1400 nM T20251 CV19HQ 72375835 IC50 = 6900 nM T20251 CJ9T5X 72375921 IC50 = 40000 nM T20251 CCP0Q4 72376019 IC50 = 26000 nM T20251 C3B0CK 72544445 IC50 > 30000 nM T20251 C1A4YW 72545684 IC50 > 30000 nM T20251 CU0NH5 72546987 IC50 = 170 nM T20251 C5WXJ6 72546988 IC50 = 530 nM T20251 CBK6T9 72546989 IC50 = 290 nM T20251 CU80HY 72547065 IC50 = 10600 nM T20251 CE3X8Y 72547066 IC50 = 2300 nM T20251 CCVG84 72547070 IC50 = 4800 nM T20251 CX70JT 72547320 IC50 = 4900 nM T20251 CY19IP 72547496 IC50 = 1500 nM T20251 CO1PV2 72548922 IC50 = 980 nM T20251 C8JTK6 72549156 IC50 > 19000 nM T20251 CT0RY5 72550282 IC50 > 20000 nM T20251 C2Q6YJ 72670421 IC50 > 10000 nM T20251 CN2GV9 72697443 IC50 = 47500 nM T20251 CCT15O 72703033 IC50 = 3700 nM T20251 CPIO30 72706193 IC50 = 350 nM T20251 C1CQG9 72706253 IC50 = 9200 nM T20251 CF4W8Z 72706442 IC50 = 2200 nM T20251 CX6T7A 72706947 IC50 = 29000 nM T20251 CBE48L 72707143 IC50 > 10000 nM T20251 CRNB25 72711191 IC50 > 33000 nM T20251 C1XSU9 72711835 IC50 > 33000 nM T20251 C29YGC 72712370 IC50 = 2300 nM T20251 C7A5EW 72714054 IC50 > 20000 nM T20251 C7SZ3V 72714058 IC50 = 35300 nM T20251 C61NKZ 72720906 IC50 > 100000 nM T20251 C6PLC5 72722131 IC50 = 25900 nM T20251 C8QEJ3 72725792 IC50 > 50000 nM T20251 C7AO4X 72792633 IC50 > 33000 nM T20251 CLK7O4 72792692 IC50 > 33000 nM T20251 CO4EX3 72793304 IC50 = 4080 nM T20251 C0KWR6 72793305 IC50 = 40 nM T20251 C65WZH 72793306 Ki = 1.8 nM T20251 C7YIT5 72793307 IC50 = 7820 nM T20251 CQ0S4C 72793308 IC50 = 3543 nM T20251 CU19BY 72793309 IC50 = 2654 nM T20251 CY42BM 72793378 IC50 = 4.9 nM T20251 C9IHR7 72793379 IC50 = 3470 nM T20251 CM04AY 72793380 IC50 = 5090 nM T20251 CTD8U0 72793381 Ki = 97 nM T20251 C0J2HG 72793383 IC50 = 4394 nM T20251 CW3O4P 72793384 IC50 = 6007 nM T20251 C6VC4N 72793385 IC50 = 53 nM T20251 CJ8RX9 72793386 IC50 = 5590 nM T20251 C6D9FH 72793441 IC50 = 1890 nM T20251 C5IL8C 72793442 IC50 = 473 nM T20251 CMK6T0 72793446 IC50 = 7372 nM T20251 CD5W8J 72793447 IC50 = 834 nM T20251 CPS57O 72793448 IC50 = 4810 nM T20251 C5BX1R 72793512 IC50 = 970 nM T20251 CHG41A 72793513 IC50 = 1050 nM T20251 C9AUO5 72793514 IC50 = 243 nM T20251 CQJF87 72793517 IC50 = 1127 nM T20251 CD5O1Q 72793518 IC50 < 5 nM T20251 C24KXZ 72793520 Ki = 119 nM T20251 CN7R9Y 72793578 IC50 = 1868 nM T20251 CZ57PR 72793579 IC50 = 238 nM T20251 C16GMC 72793580 IC50 = 1178 nM T20251 C13QTN 72793581 IC50 = 1.5 nM T20251 CB4CT7 72793582 IC50 = 2500 nM T20251 CWGK78 72793583 IC50 = 123 nM T20251 CH07SV 72793584 IC50 = 124 nM T20251 CHDB60 72793898 IC50 = 3200 nM T20251 C6R8DI 72943374 IC50 > 50000 nM T20251 C6ZA8H 72945087 IC50 > 10000 nM T20251 C7MS4G 72945112 IC50 = 13100 nM T20251 CXOI39 72945311 IC50 = 4600 nM T20251 C5TS1M 72945313 IC50 = 1000 nM T20251 CH63BO 72945314 IC50 = 700 nM T20251 C2VU8F 72945510 IC50 = 2400 nM T20251 CQ5MD0 72945512 IC50 = 3800 nM T20251 C4EM1B 72945827 IC50 > 50000 nM T20251 C1G5DP 72945830 IC50 > 50000 nM T20251 C8RLE2 72946008 IC50 > 50000 nM T20251 CDG6A2 72946010 IC50 > 50000 nM T20251 C3N7RS 72946013 IC50 = 49600 nM T20251 COEL45 72946092 IC50 > 30000 nM T20251 C37UZP 72946198 IC50 > 50000 nM T20251 CF65HX 72946199 IC50 > 50000 nM T20251 CI8Z0Q 72946200 IC50 > 50000 nM T20251 C9FLS6 72946202 IC50 = 42600 nM T20251 CA4L5S 72946204 IC50 > 50000 nM T20251 CPA9G7 72946205 IC50 = 42100 nM T20251 CF7WR3 72946381 IC50 > 50000 nM T20251 CX82VR 72946384 IC50 > 50000 nM T20251 C7X2ZL 72946387 IC50 > 50000 nM T20251 C16RLM 72946775 IC50 > 50000 nM T20251 CP21YZ 72946982 IC50 > 50000 nM T20251 CB51JH 72947191 IC50 > 50000 nM T20251 CZR9S4 72947193 IC50 > 50000 nM T20251 CMB52G 72947411 IC50 = 24100 nM T20251 CN8U7J 72947413 IC50 > 50000 nM T20251 CU9NB5 72947593 IC50 > 50000 nM T20251 C7TIG1 72947595 IC50 > 50000 nM T20251 CJQ04K 72948000 IC50 > 50000 nM T20251 CO42FH 72948001 IC50 > 50000 nM T20251 CFC70R 72948004 IC50 > 50000 nM T20251 CR70EY 72948808 IC50 = 37000 nM T20251 CA76TR 72948995 IC50 = 63400 nM T20251 CDN18F 72950534 IC50 = 109.1 nM T20251 C8R1CQ 72950535 IC50 = 416.8 nM T20251 CJZW17 72950698 IC50 = 216 nM T20251 CQF4K5 72950786 IC50 = 1000 nM T20251 C9WU2M 72950813 IC50 > 20000 nM T20251 CY9A0D 73211784 IC50 > 10000 nM T20251 CH1JK9 73213123 EC50 > 50000 nM T20251 C62TJC 73254853 EC50 > 30000 nM T20251 CG8RI0 73292361 IC50 = 7100 nM T20251 CBQ72N 73292545 IC50 = 9100 nM T20251 CKA79H 73292924 IC50 = 20000 nM T20251 C95JUO 73293105 IC50 = 600 nM T20251 CRY7G9 73294187 IC50 = 1500 nM T20251 CQV1P0 73294507 IC50 = 4200 nM T20251 C7EW4M 73294791 IC50 = 7330 nM T20251 C31ZVM 73294948 IC50 > 10000 nM T20251 CV2B0K 73294950 IC50 > 10000 nM T20251 CG8T3O 73295804 IC50 > 10000 nM T20251 CG9L2Q 73295805 IC50 > 30000 nM T20251 C5F0XZ 73295967 IC50 > 10000 nM T20251 C46HKB 73295968 IC50 > 10000 nM T20251 CTP8H1 73296128 IC50 > 10000 nM T20251 C7S0QC 73296291 IC50 > 10000 nM T20251 C86WRD 73296431 IC50 > 10000 nM T20251 C7G5OI 73296435 IC50 > 10000 nM T20251 C59TYH 73296577 IC50 > 10000 nM T20251 C9LBA7 73296578 IC50 > 10000 nM T20251 CWJS76 73331695 IC50 > 30000 nM T20251 C57LGA 73349098 IC50 = 44000 nM T20251 CX08AE 73349556 IC50 = 418350 nM T20251 CC5B9P 73351121 IC50 = 18660 nM T20251 CT1XL6 73352589 IC50 = 131 nM T20251 C3EV2U 73352607 IC50 = 5600 nM T20251 CG7R3F 73353420 IC50 = 13000 nM T20251 C0K7WP 73356819 IC50 = 206000 nM T20251 C5LBH4 73357152 IC50 = 42970 nM T20251 C6AN3L 73357170 IC50 = 11 nM T20251 C9ODB8 73387740 IC50 > 30000 nM T20251 CT1E6V 73387743 IC50 = 17300 nM T20251 CU3D9N 73388373 EC50 = 39810.72 nM T20251 CRA5H6 73389570 IC50 > 10000 nM T20251 C6V2TF 73426595 IC50 = 30000 nM T20251 C8JTD0 73442848 IC50 > 60000 nM T20251 CEP9F4 73507167 IC50 = 15800 nM T20251 CVF5P0 73603034 IC50 = 2700 nM T20251 C1SD9O 73670857 IC50 = 300 nM T20251 CJQ8B4 73670858 IC50 = 230 nM T20251 CM3Y6X 73670970 EC50 > 30000 nM T20251 CC3AG1 73670971 EC50 > 30000 nM T20251 C06YDA 73671018 IC50 = 2540 nM T20251 CJOU70 73671602 IC50 = 7200 nM T20251 CNIL19 73671824 IC50 = 1570 nM T20251 C85GVU 73671825 IC50 = 4530 nM T20251 C2K5DS 73672762 IC50 = 1900 nM T20251 C5XM3C 73673377 IC50 = 20 nM T20251 CYX59S 73673505 IC50 > 100000 nM T20251 CGC10B 73777172 IC50 = 6309.57 nM T20251 C5LPC2 73777186 IC50 = 3981.07 nM T20251 C3NDE7 73777188 IC50 = 12589.25 nM T20251 CS71JA 73777210 IC50 = 10000 nM T20251 CK3W5O 73777215 IC50 = 7943.28 nM T20251 CJ86QT 73953235 IC50 = 10000 nM T20251 CMU19S 74221664 IC50 > 30000 nM T20251 CZ3TB5 74221949 IC50 = 64000 nM T20251 CW9N8T 74222036 IC50 = 74000 nM T20251 CZK27X 74627726 IC50 = 26 nM T20251 C7M4FR 75201717 IC50 = 36000 nM T20251 C0OJ7W 75201718 IC50 = 16000 nM T20251 C2S0CO 75201720 IC50 > 80000 nM T20251 C5S2HO 75201785 IC50 = 16000 nM T20251 C4U5MR 75201786 IC50 = 6700 nM T20251 C6S2ZO 75201851 IC50 = 43000 nM T20251 C2E7QW 75201901 IC50 = 12000 nM T20251 CPS18J 75276948 EC50 > 80000 nM T20251 CF1G7P 76070567 IC50 = 3490 nM T20251 CW61JI 76071739 IC50 = 13200 nM T20251 C1W9RS 76072334 IC50 > 10000 nM T20251 CQ71AT 76073628 IC50 = 1700 nM T20251 C0N3RW 76282073 IC50 > 30000 nM T20251 CN2M8A 76284154 IC50 = 7300 nM T20251 C5ALQ2 76285468 IC50 > 10000 nM T20251 CFRU64 76285722 IC50 > 30000 nM T20251 C52KTI 76286498 IC50 = 9300 nM T20251 CZF0N7 76287389 IC50 > 30000 nM T20251 CDM04P 76310604 IC50 = 3960 nM T20251 C18SIP 76310732 IC50 = 8500 nM T20251 CO1TF8 76311072 IC50 = 30000 nM T20251 CL3N7Y 76311099 IC50 < 10 nM T20251 CB2QY6 76311111 IC50 > 33000 nM T20251 CY43DL 76311112 IC50 > 33000 nM T20251 CMF40L 76313439 IC50 = 400 nM T20251 CT2QF9 76314234 IC50 > 50000 nM T20251 CA83KU 76314239 IC50 = 2340 nM T20251 CSFB37 76314242 IC50 = 22900 nM T20251 CJ38IO 76314519 EC50 = 9800 nM T20251 C8HIS3 76314722 IC50 > 33000 nM T20251 C7K2WL 76314723 IC50 > 33000 nM T20251 C1H0GX 76314724 IC50 > 33000 nM T20251 CSL9B8 76317193 Ki > 10000 nM T20251 CEUN37 76317941 IC50 = 2000 nM T20251 CN8Q6E 76318296 IC50 > 33000 nM T20251 C1ZY4T 76318298 IC50 > 33000 nM T20251 CET31O 76318342 IC50 = 176600 nM T20251 CCMW30 76320680 IC50 = 1400 nM T20251 CDE3Y9 76321032 IC50 = 4000 nM T20251 C3TXQ5 76321521 IC50 = 16800 nM T20251 CQT3F1 76321527 IC50 > 50000 nM T20251 CEK3O5 76321713 IC50 = 6000 nM T20251 CNY2D6 76321910 EC50 = 20000 nM T20251 CR05PL 76322043 IC50 = 6100 nM T20251 CQ3CW1 76322044 IC50 = 12000 nM T20251 CYXU43 76322162 IC50 > 100000 nM T20251 C8N9QM 76325121 IC50 > 50000 nM T20251 CD3CE2 76325259 IC50 = 2800 nM T20251 CC79HT 76325260 IC50 = 6800 nM T20251 CHDF36 76325614 IC50 > 33000 nM T20251 CS27NF 76325615 IC50 > 33000 nM T20251 C3C7HE 76325645 IC50 = 48000 nM T20251 C2HCL6 76327886 IC50 = 200 nM T20251 CP9V7B 76328692 IC50 = 1260 nM T20251 CI3U1S 76328815 IC50 = 2700 nM T20251 CF27TB 76328817 IC50 = 1800 nM T20251 C5UMK8 76328829 IC50 > 40000 nM T20251 C8CQ9Y 76328873 IC50 = 14000 nM T20251 C8H9JD 76329183 IC50 > 33000 nM T20251 CAXT31 76329184 IC50 > 33000 nM T20251 C7S0CZ 76329185 IC50 > 33000 nM T20251 CWD5R4 76331595 IC50 = 3 nM T20251 CS7MR5 76331825 IC50 = 58 nM T20251 C2YIP6 76332364 IC50 = 12500 nM T20251 CNA06U 76332366 IC50 = 780 nM T20251 CI2K3T 76332845 IC50 > 33000 nM T20251 CTVI40 76332894 IC50 = 4000 nM T20251 CL7TN0 76332895 IC50 = 5600 nM T20251 CZ93JC 76335400 IC50 = 14443 nM T20251 C3Y0WL 76335990 IC50 > 50000 nM T20251 CGE5S3 76336366 EC50 = 32000 nM T20251 C0VAU9 76336449 IC50 < 10 nM T20251 CD7TI2 76336464 IC50 > 33000 nM T20251 C92WBQ 76336500 IC50 = 12700 nM T20251 C8KBZ1 76336501 IC50 = 1500 nM T20251 CQM69X 76336502 IC50 = 23300 nM T20251 C5PW6K 76683678 IC50 > 10000 nM T20251 CXM51U 76683680 IC50 = 4900 nM T20251 CGE15Z 76683773 IC50 > 10000 nM T20251 CL03DO 76683775 IC50 > 10000 nM T20251 C8HAR3 76683777 IC50 > 10000 nM T20251 CG0TR9 76683781 IC50 = 2200 nM T20251 C95OWP 76683875 IC50 = 3900 nM T20251 C67SLP 76683883 IC50 > 10000 nM T20251 C6IS1X 76683885 IC50 > 10000 nM T20251 CBSD29 76683976 IC50 > 10000 nM T20251 C0WR4O 76684092 IC50 > 10000 nM T20251 CR76SA 76684100 IC50 > 10000 nM T20251 CLD49W 76684104 IC50 = 3100 nM T20251 C08EZV 76684202 IC50 > 10000 nM T20251 C75VCS 76684206 IC50 > 10000 nM T20251 CKC14S 76684208 IC50 > 10000 nM T20251 CV62NT 76684214 IC50 = 5200 nM T20251 C8P7EC 76684296 IC50 = 2200 nM T20251 C6MSH2 76684391 IC50 > 10000 nM T20251 CAT95V 76685067 IC50 = 79750 nM T20251 CR3N1A 76900049 IC50 > 40000 nM T20251 CM73EU 76901852 IC50 = 14800 nM T20251 CQT14W 76955651 IC50 = 10100 nM T20251 C9EP7I 77003908 IC50 > 10000 nM T20251 C51DJB 77050686 IC50 > 10000 nM T20251 C2JTH8 77107528 IC50 > 30000 nM T20251 CPZ92R 77460996 IC50 = 140 nM T20251 C34TAM 77845572 IC50 > 30000 nM T20251 CT6E4H 77846842 IC50 = 700 nM T20251 CX5A7E 77846926 IC50 > 10000 nM T20251 CLC6F8 77938792 IC50 = 6400 nM T20251 CAV9J0 77989921 IC50 = 3600 nM T20251 CQZ0L8 78158242 IC50 >= 10000 nM T20251 C2NCH9 78318214 IC50 > 30000 nM T20251 C2GET7 78318815 IC50 > 30000 nM T20251 CKOU34 78319724 IC50 = 3900 nM T20251 CO0DA2 78320170 IC50 = 10800 nM T20251 C5FP1U 78321115 IC50 > 100000 nM T20251 C43NLO 78322060 IC50 = 9870 nM T20251 CV0P3A 78357783 IC50 = 14800 nM T20251 CDX94E 78426574 IC50 = 5600 nM T20251 C86QLE 81689770 IC50 = 8000 nM T20251 C9GQS2 81689815 IC50 = 50000 nM T20251 C3U0KE 81689842 IC50 > 100000 nM T20251 CHW72V 82556507 IC50 > 25000 nM T20251 CQ74UP 84626694 IC50 = 41000 nM T20251 CQMB31 85470872 IC50 > 10000 nM T20251 CLG83C 86268944 IC50 > 20000 nM T20251 CA1CE3 86270720 IC50 > 10000 nM T20251 C9TE7X 86271008 IC50 > 10000 nM T20251 CMZV56 86271009 IC50 > 10000 nM T20251 CXN93A 86271108 IC50 > 10000 nM T20251 CZL23E 86271138 IC50 > 100000 nM T20251 C5IR2K 86271238 IC50 = 8500 nM T20251 CN9MO7 86271494 IC50 > 3000 nM T20251 C4T3IW 86272102 IC50 = 39000 nM T20251 C30NBD 86272865 IC50 = 12589.25 nM T20251 C3OLB1 86274489 IC50 = 66000 nM T20251 CAB78T 86274732 IC50 = 50000 nM T20251 CCU13T 86275207 IC50 = 50000 nM T20251 CMR27C 86276168 IC50 > 25000 nM T20251 COS71Y 86276169 IC50 > 25000 nM T20251 CK20QY 86276216 IC50 > 100000 nM T20251 CW0ER2 86276224 IC50 = 900 nM T20251 CF4QX9 86278359 IC50 > 10000 nM T20251 CL09JQ 86279005 IC50 = 19560 nM T20251 CQC9M3 86279081 IC50 = 1000 nM T20251 C98IVM 86279102 Ki = 3300 nM T20251 CFJ10Z 86279104 Ki = 28800 nM T20251 CI5N8M 86279145 IC50 = 1200 nM T20251 CXF9Q3 86279146 IC50 = 10000 nM T20251 C4Y3VP 86279147 IC50 > 33000 nM T20251 CSL0I1 86279148 IC50 > 33000 nM T20251 CU70DL 86279235 IC50 = 3600 nM T20251 C38CMG 86279412 IC50 > 10000 nM T20251 C31OGJ 86279928 IC50 > 20000 nM T20251 CH3FN8 86288905 IC50 = 6800 nM T20251 CO74AR 86292101 IC50 = 5000 nM T20251 CF7GZ5 86292750 IC50 = 20800 nM T20251 CF7Y2I 86292753 IC50 = 2600 nM T20251 CV8OI5 86292754 IC50 = 1430 nM T20251 CDV37Y 86292938 IC50 = 15000 nM T20251 CZ97VP 86294733 IC50 = 24900 nM T20251 CN0W9I 86302543 IC50 = 600 nM T20251 C9EMQ0 86304601 IC50 > 30000 nM T20251 C5ZI4L 86341927 EC50 = 22800 nM T20251 CZI4Q8 86342076 EC50 > 30000 nM T20251 C4EQ8X 86342079 EC50 = 14100 nM T20251 CMK19R 86342113 EC50 > 30000 nM T20251 C73LNE 86342141 EC50 = 18800 nM T20251 CK03YC 86342156 IC50 = 2110 nM T20251 CB5F1W 86343364 IC50 = 2100 nM T20251 CKG7N2 86343365 IC50 = 13800 nM T20251 C9IVM5 86343366 IC50 = 4800 nM T20251 CMXZ65 86346192 IC50 > 50000 nM T20251 C6CD1Z 86617892 IC50 > 32000 nM T20251 CH86IJ 86670613 IC50 > 80000 nM T20251 CMG39E 86673884 IC50 > 30000 nM T20251 C9NTP1 86677234 IC50 = 5600 nM T20251 C5YX8T 86677253 IC50 = 15600 nM T20251 CCX1U5 86677265 IC50 = 7400 nM T20251 CZQ1F7 86677270 IC50 = 4300 nM T20251 CDXM47 86677874 IC50 = 75000 nM T20251 CXJA65 86685547 IC50 = 10000 nM T20251 CTG76E 86687532 IC50 > 30000 nM T20251 CR76VN 86694482 IC50 = 1200 nM T20251 CRJ9F2 86699098 IC50 > 72000 nM T20251 C52BXE 86705377 IC50 = 490 nM T20251 CC8I0M 86707711 IC50 = 3000 nM T20251 CMK52I 86721807 Ki = 780 nM T20251 CZ5J3N 86721820 Ki = 1800 nM T20251 COA34E 86721822 Ki = 1300 nM T20251 CNDS02 86722641 IC50 = 8800 nM T20251 CS7T2Z 86722660 IC50 = 8600 nM T20251 CVJ8L5 86728666 IC50 = 3500 nM T20251 C3FE1T 86730519 IC50 = 6500 nM T20251 CJ0V5L 86730522 IC50 = 2100 nM T20251 CA17UE 86732669 IC50 > 30000 nM T20251 C7OIC6 86762648 IC50 = 4300 nM T20251 CQ45XR 86763358 IC50 > 3162.28 nM T20251 CF70JO 86765186 IC50 = 12870 nM T20251 CR7Y9T 86766090 IC50 = 4500 nM T20251 C2U0BG 87055263 IC50 = 4600 nM T20251 C02UGP 87056204 IC50 = 24000 nM T20251 C6FO9E 87152177 IC50 = 13000 nM T20251 CNVS32 87343636 IC50 > 30000 nM T20251 C2EMU3 87509467 IC50 = 1132 nM T20251 CH7N2Y 87509988 IC50 = 2862 nM T20251 CF67AV 88875879 IC50 > 30000 nM T20251 C7QJ8S 88886827 IC50 = 24000 nM T20251 C6JLC2 89315866 IC50 = 1600 nM T20251 CWR09T 89449220 IC50 = 1800 nM T20251 CTC40E 89449230 IC50 = 6400 nM T20251 CW4Z2F 89470642 IC50 = 40000 nM T20251 CBRF87 89470690 IC50 > 60000 nM T20251 C7B8OH 89470730 IC50 > 60000 nM T20251 CHUO79 89471082 IC50 > 60000 nM T20251 CDQ8C6 89471114 IC50 = 40000 nM T20251 C4G5LP 89471136 IC50 > 60000 nM T20251 CX1DZ3 89471497 IC50 = 32000 nM T20251 CX1MA3 89471556 IC50 = 26000 nM T20251 CGY2Z5 89486768 IC50 = 1600 nM T20251 CQCJ02 89512686 Ki > 10000 nM T20251 C1CR9M 89512731 Ki = 2950 nM T20251 CTE1L0 89517065 IC50 = 1600 nM T20251 C56KSC 89517226 IC50 = 26000 nM T20251 CP8X3E 89573118 IC50 > 10000 nM T20251 C71QCV 89582842 Ki = 4100 nM T20251 C47HED 89583208 IC50 > 10000 nM T20251 C83JRE 89583782 IC50 > 60000 nM T20251 C1ZPE2 89583933 IC50 = 2100 nM T20251 CU74LB 89584002 IC50 = 3300 nM T20251 CBQ8J0 89584012 IC50 = 5300 nM T20251 CR0P6K 89584034 IC50 = 9100 nM T20251 C4NZW1 89584050 IC50 = 3300 nM T20251 CZOJ21 89584118 IC50 = 19000 nM T20251 CC94YO 89584863 Ki = 3800 nM T20251 CNZ2I8 89584875 Ki = 26900 nM T20251 CIBL54 89584906 Ki = 3000 nM T20251 CQY4J1 89584935 Ki = 19000 nM T20251 CP4T5E 89619103 IC50 = 5900 nM T20251 C89MLI 89619107 IC50 = 10000 nM T20251 CZ1A3U 89619266 IC50 = 12300 nM T20251 C7T9GQ 89633340 IC50 = 75900 nM T20251 C4D3MX 89633347 IC50 = 41500 nM T20251 CXPV63 89633380 IC50 = 10000 nM T20251 CRWG69 89633382 IC50 > 10000 nM T20251 CX4MP3 89633392 IC50 > 90000 nM T20251 C5FZ4E 89633466 IC50 = 33700 nM T20251 CX90VG 89691439 IC50 > 10000 nM T20251 CXR3A4 89702226 IC50 > 10000 nM T20251 CA49UY 89726151 IC50 > 10000 nM T20251 CIXB02 89738547 IC50 > 10000 nM T20251 C9X3MF 89752438 IC50 = 7600 nM T20251 CF5RQ7 89762819 IC50 = 18000 nM T20251 C8MN9K 89763714 IC50 = 1100 nM T20251 C5MR9K 89777151 IC50 > 33000 nM T20251 CI57QV 89782019 IC50 > 30000 nM T20251 C7TRY9 89844945 IC50 > 80000 nM T20251 CE2Z4C 89845025 IC50 > 80000 nM T20251 CTP94N 89845031 IC50 > 80000 nM T20251 C5RAI0 89907349 IC50 = 17000 nM T20251 CP0GY3 89908140 IC50 = 1800 nM T20251 C0JA2V 89908303 IC50 = 1500 nM T20251 CJW7L6 89908440 IC50 > 30000 nM T20251 CN76VK 89912923 IC50 = 15848.93 nM T20251 C2MPT3 89954418 IC50 > 10000 nM T20251 C54XDY 89975061 IC50 = 110 nM T20251 C5YEP2 89992279 IC50 = 4900 nM T20251 C8P1SX 89992280 IC50 > 10000 nM T20251 C0R6LF 89992295 IC50 = 3200 nM T20251 C63CJN 89992309 IC50 = 8900 nM T20251 CQ5HZ7 89996234 IC50 > 30000 nM T20251 CAKV98 89997377 Ki > 10000 nM T20251 CIBY41 89997417 Ki = 11700 nM T20251 C8Z9QB 89997423 Ki = 2950 nM T20251 C4PT6B 89997503 Ki > 10000 nM T20251 CB7L1N 89997512 Ki > 10000 nM T20251 CE7PH6 89997520 Ki > 10000 nM T20251 C52QPK 89997526 Ki = 145 nM T20251 C90TSY 89997709 Ki > 15000 nM T20251 C2SJY8 89997744 Ki > 10000 nM T20251 CFYO09 89997799 Ki > 10000 nM T20251 C7Z1GY 89997802 Ki > 15000 nM T20251 C89LAZ 89997856 Ki > 15000 nM T20251 C5EQM4 89997906 Ki = 377 nM T20251 C7M5KB 89997911 Ki > 15000 nM T20251 CXP2Q5 89997939 Ki = 797 nM T20251 CX4S6M 89997948 Ki = 90 nM T20251 COR4F3 89997978 Ki > 15000 nM T20251 CDI4P0 89997990 Ki > 15000 nM T20251 C9TG4Q 89998018 Ki > 10000 nM T20251 CN0DA6 89998034 Ki = 210 nM T20251 CD1VM9 89998106 Ki > 10000 nM T20251 CT38QK 89998122 Ki > 10000 nM T20251 CMO1B0 89998184 Ki = 259 nM T20251 CZ5QN1 89998216 Ki = 3810 nM T20251 C7NA0W 89998237 Ki > 10000 nM T20251 CRTP06 90000797 IC50 > 30000 nM T20251 C0NM2P 90001216 IC50 > 30000 nM T20251 C1RDQ2 90043471 IC50 > 30000 nM T20251 C3CYP0 90043482 IC50 > 30000 nM T20251 CAM93E 90043622 IC50 > 10000 nM T20251 CJ4KS1 90043633 IC50 > 10000 nM T20251 CY82BX 90044129 IC50 > 30000 nM T20251 CG5P9A 90153688 IC50 = 2500 nM T20251 CV6H7R 90153809 IC50 = 38000 nM T20251 CE7N6F 90265032 IC50 = 16600 nM T20251 C0M7NI 90268057 IC50 = 1551 nM T20251 CY5P6I 90268061 IC50 = 16940 nM T20251 CP0X1V 90311949 IC50 = 14400 nM T20251 C75FLG 90326903 IC50 = 19700 nM T20251 C26LKW 90341025 IC50 > 30000 nM T20251 C9UZX2 90355303 IC50 = 1700 nM T20251 CTO87I 90355486 IC50 = 8500 nM T20251 CB1P9Y 90355676 IC50 = 2400 nM T20251 C03ZXF 90355716 IC50 = 17700 nM T20251 CDN1X8 90366524 IC50 = 6100 nM T20251 CTV52A 90367281 IC50 = 3000 nM T20251 CA47VK 90408538 IC50 > 10000 nM T20251 CE4IT5 90408860 IC50 > 3000 nM T20251 CB0RP3 90410604 IC50 > 10000 nM T20251 CQ8ZW3 90410911 IC50 > 10000 nM T20251 CD5W6K 90417914 IC50 = 7300 nM T20251 CDJ1R8 90418278 IC50 > 50000 nM T20251 CV9HL2 90420193 IC50 = 15000 nM T20251 CTZY03 90420346 IC50 > 11000 nM T20251 C1X7PZ 90420407 IC50 = 2900 nM T20251 CX3AU6 90420765 IC50 > 33000 nM T20251 CL4WR9 90465846 IC50 = 11700 nM T20251 CJE7P5 90467013 IC50 > 33000 nM T20251 CX6DQ4 90467014 IC50 > 33000 nM T20251 C7D2UK 90467156 IC50 > 33000 nM T20251 CV75ZC 90467159 IC50 > 33000 nM T20251 C3RO1M 90467162 IC50 > 33000 nM T20251 C6BID5 90469437 IC50 > 10000 nM T20251 CW61DN 90488999 IC50 = 7400 nM T20251 CF30KA 90643570 IC50 = 31000 nM T20251 C2CE9A 90643781 Ki = 2000 nM T20251 C05MTO 90643782 Ki = 620 nM T20251 C6RM2B 90643783 Ki > 10000 nM T20251 CPD10X 90643784 Ki > 10000 nM T20251 CUB0Q1 90643785 Ki > 10000 nM T20251 CPN65E 90643787 IC50 > 30000 nM T20251 C1HGB2 90644097 IC50 = 5300 nM T20251 C83UOX 90644098 IC50 = 26000 nM T20251 C3BM4E 90644099 IC50 = 69000 nM T20251 C5VTU0 90644100 IC50 = 50600 nM T20251 CICV18 90644101 IC50 = 10000 nM T20251 CIM7G0 90644102 IC50 = 33000 nM T20251 CFB56D 90644103 IC50 = 2500 nM T20251 C1D4UG 90644104 IC50 = 74000 nM T20251 CV0X9O 90644105 IC50 = 12000 nM T20251 C8Y2XF 90644106 IC50 = 69000 nM T20251 CG48ID 90644107 IC50 = 13000 nM T20251 CZ8BP9 90644108 IC50 > 100000 nM T20251 CKAB34 90644109 IC50 > 100000 nM T20251 C13AEC 90644110 IC50 = 133000 nM T20251 C87MOQ 90644111 IC50 = 90000 nM T20251 CUK9C4 90644112 IC50 = 151000 nM T20251 CW7K6S 90644113 IC50 > 100000 nM T20251 CQJ1C8 90644114 IC50 > 100000 nM T20251 C4MHY0 90644115 IC50 > 100000 nM T20251 C6TR0K 90644116 IC50 > 100000 nM T20251 CCJQ83 90644117 IC50 > 100000 nM T20251 C3JMQ9 90644367 IC50 = 2750 nM T20251 CMV2F4 90644368 IC50 = 17000 nM T20251 CGN7C6 90644461 IC50 > 100000 nM T20251 C7R3QG 90644462 IC50 > 100000 nM T20251 CI62FU 90644463 IC50 > 100000 nM T20251 C9R6LO 90644464 IC50 > 33000 nM T20251 C8TK5D 90644465 IC50 = 16000 nM T20251 CBT08V 90644466 IC50 > 33000 nM T20251 CU9K6R 90644467 IC50 > 33000 nM T20251 CB12SV 90644468 IC50 > 33000 nM T20251 C7WIM0 90644678 IC50 = 18000 nM T20251 C5O8HN 90644762 IC50 > 10500 nM T20251 CZ5YK9 90644763 IC50 > 33300 nM T20251 CUK5T1 90644764 IC50 > 33300 nM T20251 CIHE96 90644765 IC50 > 33300 nM T20251 CY4PB3 90644766 IC50 > 33300 nM T20251 CVUE08 90644767 IC50 > 33300 nM T20251 CV79BJ 90644768 IC50 > 33300 nM T20251 CL5UB3 90644769 IC50 > 33300 nM T20251 C6AMK9 90644770 IC50 = 16600 nM T20251 CK84IG 90644771 IC50 = 3500 nM T20251 CQVY70 90644772 IC50 = 4500 nM T20251 CAVN86 90644773 IC50 = 12200 nM T20251 CPS9I2 90644774 IC50 = 10300 nM T20251 C1VU8Q 90644775 IC50 = 22000 nM T20251 CMQ30B 90644776 IC50 = 25000 nM T20251 C6FL9K 90644777 IC50 > 33300 nM T20251 CXSJ16 90644778 IC50 > 33300 nM T20251 CV3C5H 90644779 IC50 = 60000 nM T20251 C0KQV4 90645474 IC50 = 135 nM T20251 CE8AI2 90654467 IC50 = 920 nM T20251 CV87PR 90655950 IC50 > 40000 nM T20251 C62SML 90655967 IC50 > 33000 nM T20251 CJ7LT3 90655968 IC50 > 33000 nM T20251 CB61WC 90655969 IC50 > 33000 nM T20251 CK6QN4 90656025 IC50 > 50000 nM T20251 CO73FL 90656026 IC50 > 50000 nM T20251 COW7U5 90656027 IC50 = 3100 nM T20251 CV9H8U 90656285 IC50 > 30000 nM T20251 CDF9O2 90656287 IC50 = 8200 nM T20251 CIL2W9 90664452 IC50 = 9800 nM T20251 C4MUI2 90664601 IC50 = 8110 nM T20251 CA79EY 90664683 IC50 = 1700 nM T20251 CTR58M 90664931 IC50 = 1000 nM T20251 CHT7D5 90664962 IC50 > 10000 nM T20251 C01UNB 90665166 Ki = 3760 nM T20251 CXJ62T 90665173 IC50 = 900 nM T20251 CG98QO 90665194 IC50 = 1300 nM T20251 CJCR26 90665456 IC50 = 9670 nM T20251 C71ARQ 90665737 IC50 = 22000 nM T20251 CZOW03 90665738 IC50 = 4000 nM T20251 CVJE69 90665739 IC50 = 59000 nM T20251 CG4E8W 90665845 IC50 = 8700 nM T20251 C1S7YU 90665846 IC50 = 2100 nM T20251 C8B1RN 90665847 IC50 = 3500 nM T20251 CCQ67W 90665848 IC50 = 2100 nM T20251 C2DF8V 90665849 IC50 = 3700 nM T20251 CGB7U8 90665850 IC50 = 2500 nM T20251 C67YNO 90665851 IC50 > 10000 nM T20251 C2E6NI 90665852 IC50 > 8300 nM T20251 C1X2PV 90665949 IC50 = 18000 nM T20251 CKY18S 90665950 IC50 > 28000 nM T20251 CDQ56W 90665987 IC50 > 10000 nM T20251 C97PUB 90666011 IC50 = 11000 nM T20251 CU9OP3 90666012 IC50 = 10000 nM T20251 C8O2ZM 90666013 IC50 = 15000 nM T20251 C3ND7I 90666014 IC50 = 22000 nM T20251 CSJE46 90666015 IC50 = 21000 nM T20251 C6W4GH 90666017 IC50 = 47000 nM T20251 C0D5FT 90666018 IC50 = 43000 nM T20251 CMX8H0 90666019 IC50 > 100000 nM T20251 C4AP0G 90666024 IC50 = 44000 nM T20251 C5WQN4 90666035 IC50 = 2900 nM T20251 C85AMH 90666036 IC50 = 3200 nM T20251 CKF14A 90666037 IC50 = 12000 nM T20251 CM7ED5 90666038 IC50 = 4100 nM T20251 CU2T3C 90666039 IC50 = 14000 nM T20251 C59YXE 90666040 IC50 = 7300 nM T20251 C6QZL4 90666041 IC50 = 6800 nM T20251 CY35OV 90666042 IC50 = 8400 nM T20251 C2IN9R 90666094 IC50 = 1970 nM T20251 CMU2J7 90666098 IC50 = 1700 nM T20251 CU9MV6 90666148 IC50 = 18000 nM T20251 CC07QH 90666256 IC50 = 1200 nM T20251 C6H5CY 90666260 IC50 = 1900 nM T20251 C45NLU 90666267 IC50 = 1700 nM T20251 C5VZC6 90666479 IC50 = 2200 nM T20251 CQ23WR 90667215 IC50 = 13000 nM T20251 CGP3C6 90667419 IC50 = 18300 nM T20251 CF6MO3 90667420 IC50 = 1280 nM T20251 CCO96L 90667421 IC50 = 4920 nM T20251 CIW51L 90667423 IC50 = 86200 nM T20251 CG2J7Y 90667424 IC50 = 92100 nM T20251 CC7G4Q 90667584 IC50 = 210 nM T20251 CW5UZ9 90667585 IC50 = 1280 nM T20251 CGX4S0 90667586 IC50 = 390 nM T20251 CK4GF3 90667587 IC50 = 37 nM T20251 C9XVG4 90667588 IC50 = 174 nM T20251 C08COA 90667590 IC50 = 93600 nM T20251 C7BK1O 90667600 IC50 = 81700 nM T20251 CZL03G 90667602 IC50 = 107 nM T20251 CR59JY 90667603 IC50 = 75800 nM T20251 CGRK73 90667608 IC50 = 1270 nM T20251 C2ZN9Y 90667609 IC50 > 100000 nM T20251 CT5H7A 90667610 IC50 = 160 nM T20251 CTD7C6 90667611 IC50 = 480 nM T20251 CIM1S7 90667868 IC50 > 100000 nM T20251 CT2GU1 91246771 IC50 = 10700 nM T20251 CYHR27 91664373 IC50 > 10000 nM T20251 CUI10E 91666686 IC50 = 19600 nM T20251 C76AKI 91754444 IC50 = 81000 nM T20251 C7EXH8 91755097 IC50 > 80000 nM T20251 C37IZB 91755098 IC50 = 18000 nM T20251 CX4DJ7 91799322 IC50 = 800 nM T20251 C90JVH 91799688 IC50 = 49 nM T20251 CGJ6S0 91801175 IC50 > 60000 nM T20251 CK6E0W 91810397 IC50 = 48000 nM T20251 CC9B6T 91820646 IC50 = 28000 nM T20251 C3L6KU 91820689 IC50 > 40000 nM T20251 CDT6C1 91824787 Ki = 6251 nM T20251 CK5X2M 91826235 IC50 = 23000 nM T20251 C9MO7C 91826722 IC50 = 4300 nM T20251 C64QCZ 91827500 IC50 = 501.19 nM T20251 CL7S4U 91844670 IC50 > 50000 nM T20251 CSK6Z1 91844707 IC50 = 5290 nM T20251 CRX16J 91884611 IC50 = 4050 nM T20251 CBG6E7 91885506 IC50 > 10000 nM T20251 CFT9N5 91885578 IC50 = 20000 nM T20251 CU1G3S 91933941 IC50 > 30000 nM T20251 CQN41K 91938095 Ki = 1732 nM T20251 CWZX73 91971958 IC50 = 5100 nM T20251 CYMH49 92044895 IC50 > 20000 nM T20251 C38ZID 92045057 IC50 > 10000 nM T20251 CEJK10 92135927 IC50 = 21000 nM T20251 CCY0O2 100951644 IC50 > 33300 nM T20251 CNQ6J9 101873336 Ki = 7048 nM T20251 C0QXE2 101882778 IC50 = 400 nM T20251 C05NTY 101884761 IC50 = 4000 nM T20251 CWM71R 101884762 IC50 = 6700 nM T20251 C4KH1V 101886593 IC50 = 210 nM T20251 C2EJK6 101910737 IC50 = 6980 nM T20251 CB5DK1 102004349 IC50 = 400 nM T20251 CQ9PN8 102593934 IC50 > 30000 nM T20251 C4Z1OU 110451319 IC50 > 25000 nM T20251 CN57AX 110451673 IC50 > 25000 nM T20251 C8F6VO 117604931 IC50 > 100000 nM T20251 C6UOT8 117653759 IC50 = 17000 nM T20251 C8ZM9J 117678530 IC50 = 3200 nM T20251 C5CL8X 117684497 IC50 = 3500 nM T20251 C4O3VF 117689963 IC50 = 26800 nM T20251 CT7GW0 117690258 IC50 = 19700 nM T20251 CX0DY2 117690263 IC50 = 17600 nM T20251 CQF32S 117690304 IC50 = 8900 nM T20251 C15QUL 117690396 IC50 = 53400 nM T20251 CFT94I 117700435 IC50 > 10000 nM T20251 CG60JW 117700665 IC50 = 3130 nM T20251 C3GB4X 117715778 IC50 > 50000 nM T20251 C2TG7Y 117715783 IC50 = 6900 nM T20251 CW8RS3 117760464 Ki > 30000 nM T20251 CZC84D 117769161 IC50 = 10200 nM T20251 CE7BZ8 117769174 IC50 = 8500 nM T20251 CBJ07Q 117769217 IC50 > 80000 nM T20251 CXHQ08 117769229 IC50 = 7200 nM T20251 CS9WO4 117769234 IC50 = 7700 nM T20251 C1SA9I 117769244 IC50 = 35000 nM T20251 C0VY7C 117769271 IC50 = 7500 nM T20251 CSR9B0 117769289 IC50 = 5300 nM T20251 C2M9CR 117769307 IC50 = 41000 nM T20251 C7FWS3 117769309 IC50 = 12000 nM T20251 CYWV32 117769339 IC50 = 4100 nM T20251 CZV35K 117769346 IC50 > 80000 nM T20251 C5V6RG 117769349 IC50 > 80000 nM T20251 C4O1PX 117769362 IC50 = 7600 nM T20251 CPV4C8 117769365 IC50 = 13800 nM T20251 CP3MC5 117769379 IC50 = 9600 nM T20251 C8V6LG 117769392 IC50 = 8000 nM T20251 C2NBZ8 117769396 IC50 = 6000 nM T20251 COV59Y 117769408 IC50 = 4900 nM T20251 CXJ3I6 117769409 IC50 = 17000 nM T20251 C8LTZ6 117769464 IC50 > 80000 nM T20251 CSKO30 117769533 IC50 = 5000 nM T20251 C6XC3W 117769575 IC50 = 300 nM T20251 C8Y5ZX 117778486 IC50 = 9500 nM T20251 CDUH09 117809287 IC50 = 30000 nM T20251 C3FY8A 117838708 IC50 = 7800 nM T20251 C7VDL3 117838709 IC50 = 30000 nM T20251 C0BI1C 117838710 IC50 = 13500 nM T20251 CBD0X6 117852205 IC50 = 29600 nM T20251 CN5H7Y 117852210 IC50 = 7900 nM T20251 CB9X7D 117852213 IC50 = 6100 nM T20251 CTKJ90 117852221 IC50 = 1200 nM T20251 C3PST8 117852226 IC50 = 193 nM T20251 CN8G6X 117852236 IC50 = 2400 nM T20251 C3SW9X 117852238 IC50 = 3290 nM T20251 CO3X7N 117852239 IC50 > 60000 nM T20251 C17KYZ 117852241 IC50 = 17400 nM T20251 CI06AN 117852248 IC50 = 10500 nM T20251 C3K8XU 117852302 IC50 = 1800 nM T20251 CMS0A3 117852327 IC50 = 16100 nM T20251 C04UHW 117852380 IC50 = 2400 nM T20251 CQ4FJ5 117852383 IC50 = 8900 nM T20251 C0A4XC 117871929 IC50 = 2900 nM T20251 CV4B2W 117871992 IC50 > 60000 nM T20251 CY5JF0 117872250 IC50 = 6100 nM T20251 COIM28 117872315 IC50 > 60000 nM T20251 C7PM6F 117872316 IC50 = 5200 nM T20251 C6X8VS 117872368 IC50 = 40000 nM T20251 CQ5S7L 117872990 IC50 = 1900 nM T20251 C9OA4U 117873033 IC50 = 25000 nM T20251 CL6QV4 117873045 IC50 = 12000 nM T20251 C6XS8J 117887024 IC50 = 2300 nM T20251 CP0I7M 117887098 IC50 = 1200 nM T20251 CA7Z3W 117887511 IC50 = 1600 nM T20251 CFV23K 117887619 IC50 = 700 nM T20251 C89EQN 117897570 IC50 = 20200 nM T20251 C4CH7J 117955548 IC50 = 240 nM T20251 C07ACT 117955744 IC50 = 3700 nM T20251 CK53MQ 117972250 IC50 = 380 nM T20251 C9KV7L 117993993 Ki > 30000 nM T20251 CNV24M 117993998 Ki > 30000 nM T20251 CS16CJ 118022791 IC50 = 11400 nM T20251 C89WQL 118023142 IC50 = 6800 nM T20251 CFE6M2 118038416 IC50 > 10000 nM T20251 C2WQ4G 118039220 IC50 = 260 nM T20251 CTU3K2 118043167 IC50 > 10000 nM T20251 CPU7C0 118043263 IC50 = 10000 nM T20251 CR2XJ5 118043265 IC50 = 3300 nM T20251 C4HQ5C 118043312 IC50 = 1500 nM T20251 CB4A6H 118043313 IC50 > 10000 nM T20251 C45RCJ 118072307 IC50 > 80000 nM T20251 CH7LT6 118072319 IC50 > 80000 nM T20251 CUQ85I 118102658 IC50 > 30000 nM T20251 CMX3U8 118107483 IC50 = 1400 nM T20251 C5R1XP 118107577 IC50 > 10000 nM T20251 C91QJN 118107589 IC50 > 10000 nM T20251 C9JE0K 118107598 IC50 > 10000 nM T20251 C3ID1F 118111696 IC50 = 300 nM T20251 CD48WH 118121169 IC50 = 4500 nM T20251 C3F6XG 118165440 IC50 = 4000 nM T20251 CDAC50 118165497 IC50 = 6300 nM T20251 CN4O5K 118165763 IC50 = 2800 nM T20251 C0TMZ8 118167692 IC50 = 14000 nM T20251 C68QVN 118167694 IC50 = 24000 nM T20251 CSM69G 118167758 IC50 = 4200 nM T20251 C9EY8L 118167812 IC50 = 6500 nM T20251 CP8QO0 118179807 IC50 > 100000 nM T20251 CT4G5D 118179817 IC50 > 100000 nM T20251 CIU02H 118179819 IC50 = 100000 nM T20251 C4KC7H 118189484 IC50 = 9000 nM T20251 C5DYL3 118189493 IC50 = 7000 nM T20251 CLH8X7 118189551 IC50 = 9500 nM T20251 CAI09J 118195093 IC50 > 30000 nM T20251 CZ5G7W 118195200 IC50 = 4200 nM T20251 C0NM1V 118195331 IC50 = 1500 nM T20251 C3J4UQ 118198923 IC50 = 310 nM T20251 CV67TP 118207324 IC50 = 400 nM T20251 CPZ69K 118207398 IC50 > 30000 nM T20251 CG84LB 118207404 IC50 = 620 nM T20251 C1GH3R 118207538 IC50 = 7800 nM T20251 C91ECG 118217204 IC50 > 5000 nM T20251 CV16QJ 118217208 IC50 > 30000 nM T20251 CL5C4K 118253824 IC50 > 33000 nM T20251 CCH97D 118253857 IC50 = 17000 nM T20251 CCG7Y6 118253883 IC50 = 31000 nM T20251 CA72QZ 118253888 IC50 > 33000 nM T20251 CZ3U4P 118270292 IC50 = 3380 nM T20251 C3E5PL 118307312 IC50 = 3290 nM T20251 C93OPR 118307317 IC50 = 12400 nM T20251 CIY0X1 118307334 IC50 = 20100 nM T20251 CD93MJ 118307348 IC50 = 3510 nM T20251 C89TZG 118307431 IC50 > 30000 nM T20251 CKG4L3 118334971 IC50 = 2100 nM T20251 CRV14T 118334974 IC50 = 500 nM T20251 C7VYK2 118334975 IC50 = 200 nM T20251 CIS2L9 118334979 IC50 = 2000 nM T20251 CKM6L0 118334982 IC50 = 900 nM T20251 CH8PU2 118334995 IC50 = 500 nM T20251 C1TF9K 118368174 IC50 = 22000 nM T20251 CBIR89 118389918 IC50 = 15600 nM T20251 CRHY82 118409479 IC50 > 30000 nM T20251 CO75VB 118409494 IC50 > 30000 nM T20251 C3FVW7 118409564 IC50 > 30000 nM T20251 CW3IC5 118414671 IC50 = 30000 nM T20251 C94WRZ 118435363 IC50 = 9300 nM T20251 C1WL4E 118435382 IC50 = 23600 nM T20251 C5L9VH 118435403 IC50 = 12100 nM T20251 CNXH97 118435407 IC50 = 9000 nM T20251 C8Z2FP 118435412 IC50 = 10700 nM T20251 CJIP45 118435414 IC50 = 10100 nM T20251 CY6EP7 118435506 IC50 = 43000 nM T20251 CPE35X 118435524 IC50 = 9600 nM T20251 CVK6Y8 118435560 IC50 = 11700 nM T20251 CN5L8K 118435601 IC50 = 13100 nM T20251 C37SFM 118435617 IC50 = 17900 nM T20251 CZLJ20 118441559 IC50 = 400 nM T20251 CR9QF7 118441560 IC50 = 11970 nM T20251 CEMZ15 118464420 IC50 > 1000 nM T20251 CRV8S3 118478927 IC50 > 10000 nM T20251 CL32JE 118478933 IC50 > 10000 nM T20251 C5S1HZ 118478972 IC50 > 10000 nM T20251 C8G9HP 118478986 IC50 > 10000 nM T20251 CBV89G 118478994 IC50 > 10000 nM T20251 CK0ER5 118478999 IC50 > 10000 nM T20251 CU25KC 118479000 IC50 > 10000 nM T20251 CW07IS 118479006 IC50 = 6700 nM T20251 C3ZAV0 118479034 IC50 > 10000 nM T20251 C4W6ZS 118479038 IC50 > 10000 nM T20251 CRG24C 118479053 IC50 > 10000 nM T20251 CD4ME1 118479123 IC50 > 10000 nM T20251 CB0XM2 118479161 IC50 > 10000 nM T20251 C18NTQ 118479199 IC50 = 10000 nM T20251 CJ0Z1Y 118479222 IC50 > 10000 nM T20251 CP0U6Y 118479229 IC50 > 10000 nM T20251 C3A6HD 118479231 IC50 > 10000 nM T20251 CJ14CR 118479241 IC50 = 9900 nM T20251 C1FO3N 118479293 IC50 = 4300 nM T20251 CF02TZ 118479295 IC50 = 10000 nM T20251 C90TED 118479305 IC50 = 10000 nM T20251 C7I9RC 118479316 IC50 > 10000 nM T20251 CRC4F6 118479354 IC50 > 10000 nM T20251 CRCV51 118479359 IC50 > 10000 nM T20251 CJL5W0 118479428 IC50 > 10000 nM T20251 CS2VA7 118479440 IC50 > 10000 nM T20251 CJ9P0M 118479445 IC50 = 6900 nM T20251 C3U1RB 118479452 IC50 = 4500 nM T20251 CBJ28X 118483320 IC50 > 30000 nM T20251 C0KPH4 118485600 IC50 = 160 nM T20251 C43GZF 118485601 IC50 = 980 nM T20251 C8UT1Z 118485623 IC50 = 610 nM T20251 CC94IQ 118485651 IC50 = 4900 nM T20251 CMK97G 118491864 IC50 = 9000 nM T20251 C62FCZ 118491902 IC50 = 6000 nM T20251 CD57MP 118491918 IC50 > 30000 nM T20251 C05LQH 118498627 IC50 > 33000 nM T20251 CXCF46 118498683 IC50 > 33000 nM T20251 CJA07S 118498727 IC50 > 33000 nM T20251 CG6D1J 118498935 IC50 = 27000 nM T20251 CXR46C 118499887 IC50 > 33000 nM T20251 CFVN15 118500050 IC50 > 33000 nM T20251 CY9NW0 118500097 IC50 > 33000 nM T20251 CXEI18 118500108 IC50 > 33000 nM T20251 CL2Z5Y 118502821 IC50 = 22000 nM T20251 CVY64N 118502892 IC50 > 33000 nM T20251 CO20ET 118502895 IC50 = 14000 nM T20251 CU1X3H 118502919 IC50 > 33000 nM T20251 CK04PJ 118512792 IC50 = 4670 nM T20251 C48PFK 118512802 IC50 = 14500 nM T20251 C76UQN 118512804 IC50 = 1600 nM T20251 CAKI19 118514811 IC50 = 8460 nM T20251 C0R2MP 118519041 IC50 > 30000 nM T20251 CRAF61 118523357 IC50 > 33000 nM T20251 C5P7VH 118523411 IC50 = 18000 nM T20251 CD0EY5 118523423 IC50 > 33000 nM T20251 C7AYV5 118540795 Ki = 1091 nM T20251 CG19TS 118554552 IC50 > 33300 nM T20251 CU02NF 118559124 IC50 = 7570 nM T20251 CB41MH 118560618 IC50 = 5500 nM T20251 C5CDE0 118562359 IC50 = 600 nM T20251 CS63OE 118562362 IC50 = 1100 nM T20251 C60BSA 118562375 IC50 = 1200 nM T20251 CE3D0A 118562384 IC50 = 800 nM T20251 C7IVW9 118562402 IC50 = 8200 nM T20251 CE53DJ 118562440 IC50 = 600 nM T20251 CW26NV 118562451 IC50 = 300 nM T20251 C7G5HO 118562469 IC50 = 200 nM T20251 C5JKQ9 118562510 IC50 = 400 nM T20251 CF6LK7 118562538 IC50 = 1200 nM T20251 C6FOS9 118562556 IC50 = 1000 nM T20251 C25MXS 118562567 IC50 = 100 nM T20251 CJF1E6 118562576 IC50 = 100 nM T20251 C5QB2S 118562584 IC50 = 1200 nM T20251 C6TC3D 118562598 IC50 = 2000 nM T20251 CWA4B2 118562606 IC50 = 100 nM T20251 C2EPN1 118565438 IC50 = 600 nM T20251 C0XIN5 118567313 IC50 = 1900 nM T20251 C6PA1C 118567531 IC50 = 6600 nM T20251 CD4XK8 118567534 IC50 = 500 nM T20251 CLVO18 118567538 IC50 = 3300 nM T20251 C1CP6Z 118567543 IC50 > 10000 nM T20251 C32PGF 118567545 IC50 = 3800 nM T20251 C7G8IT 118567547 IC50 = 1100 nM T20251 CXW0K9 118567604 IC50 = 1200 nM T20251 C4ULH8 118567605 IC50 = 100 nM T20251 C8TP7C 118567608 IC50 = 1000 nM T20251 CI0JY2 118567747 IC50 = 1200 nM T20251 C78LNX 118572065 IC50 > 100000 nM T20251 COYJ84 118575663 IC50 > 25000 nM T20251 CSW92P 118607432 IC50 > 100000 nM T20251 CM93VO 118611725 IC50 = 8000 nM T20251 CE69HN 118613626 IC50 > 100000 nM T20251 C2EQ9X 118613653 IC50 > 100000 nM T20251 C1X8GW 118613658 IC50 > 100000 nM T20251 CVE4S5 118627059 IC50 = 1180 nM T20251 CL74GH 118665602 IC50 = 35000 nM T20251 CP71CK 118665611 IC50 = 38000 nM T20251 CR3F5V 118665613 IC50 = 29000 nM T20251 C60TWO 118665627 IC50 = 42000 nM T20251 CY7T8F 118665628 IC50 = 38000 nM T20251 CBZ59D 118701008 IC50 = 1800 nM T20251 CRS34C 118705500 IC50 > 100000 nM T20251 C2WP6X 118706538 IC50 = 1410 nM T20251 CZE4U0 118706539 IC50 = 1460 nM T20251 CP6O2R 118706799 IC50 = 190 nM T20251 C2O7GE 118707553 IC50 = 31200 nM T20251 C8S9VW 118707562 IC50 = 12900 nM T20251 C9BCT8 118707596 IC50 = 21100 nM T20251 C62JCD 118707597 IC50 = 20700 nM T20251 C8CXM5 118707599 IC50 = 22000 nM T20251 CC0VX1 118707602 IC50 = 59500 nM T20251 CN2IC3 118707603 IC50 = 19900 nM T20251 CH9MA5 118707606 IC50 = 40500 nM T20251 CRNF04 118709230 IC50 = 7000 nM T20251 CARX10 118709238 IC50 > 30000 nM T20251 CQ65IH 118709240 IC50 > 30000 nM T20251 CG96QP 118709241 IC50 = 3300 nM T20251 C8QO1J 118709242 IC50 > 30000 nM T20251 CBK73W 118709243 IC50 > 30000 nM T20251 C35GDB 118709244 IC50 > 30000 nM T20251 CI9Q7O 118709245 IC50 > 30000 nM T20251 CD0B1Z 118709246 IC50 > 30000 nM T20251 CMX6S5 118709259 IC50 > 60000 nM T20251 CM64SW 118709261 IC50 = 4800 nM T20251 C7WY2D 118709262 IC50 = 10000 nM T20251 CN25PF 118709263 IC50 = 7000 nM T20251 CU25HN 118709264 IC50 = 1000 nM T20251 CQOS43 118709267 IC50 = 1000 nM T20251 CXH06J 118709268 IC50 = 4500 nM T20251 CFZV13 118709269 IC50 = 1400 nM T20251 CTJ0H1 118709270 IC50 = 1200 nM T20251 CP9W5U 118709272 IC50 = 10000 nM T20251 C15VXF 118709274 IC50 = 1400 nM T20251 CXFS23 118709275 IC50 > 33000 nM T20251 CJ5C4D 118709276 IC50 = 2000 nM T20251 C7O1JS 118709277 IC50 = 1800 nM T20251 C1CUQ5 118709784 IC50 = 3500 nM T20251 CFN94L 118709786 IC50 = 12700 nM T20251 C32EZA 118709832 IC50 = 21500 nM T20251 CSL13X 118709837 IC50 = 7300 nM T20251 CV26JZ 118709848 IC50 = 8800 nM T20251 CFC1J5 118710523 IC50 = 707 nM T20251 C4X8NC 118710524 IC50 = 625 nM T20251 CK3WG9 118710525 IC50 = 1420 nM T20251 C4NIK8 118710526 IC50 = 1205 nM T20251 C3JAX9 118710527 IC50 = 2257 nM T20251 CXV1C5 118710528 IC50 = 2520 nM T20251 CA5TR0 118710529 IC50 = 1611 nM T20251 CX9Q7Z 118710530 IC50 = 2845 nM T20251 C27IPK 118710531 IC50 = 8703 nM T20251 C9AZ1B 118710534 IC50 = 11990 nM T20251 C0YL9Z 118710536 IC50 = 95600 nM T20251 CD34IY 118710582 IC50 = 1000 nM T20251 CYP20X 118711743 Ki = 7050 nM T20251 C47GVE 118711875 Ki = 6250 nM T20251 C2IUO5 118711883 Ki > 10000 nM T20251 C4MP7C 118711884 Ki > 10000 nM T20251 CD9E1M 118711886 Ki > 10000 nM T20251 C5A4XS 118712578 IC50 = 209000 nM T20251 CP2S6F 118712580 IC50 = 25000 nM T20251 C4T2FY 118712775 IC50 = 97700 nM T20251 C5M3BX 118712788 IC50 = 55300 nM T20251 CN4XM2 118713119 IC50 = 14000 nM T20251 C84GOU 118713773 IC50 = 4710 nM T20251 C2LY9D 118713799 IC50 = 1880 nM T20251 CMO2V7 118713801 IC50 = 5500 nM T20251 C9IXE6 118715640 IC50 = 41000 nM T20251 CMN87B 118716079 IC50 > 33000 nM T20251 CC56DO 118718808 IC50 = 56000 nM T20251 CYX8Z6 118720352 Ki = 624 nM T20251 CF5HV8 118720613 IC50 = 1500 nM T20251 C2UIB7 118720614 IC50 > 30000 nM T20251 CSH50J 118720615 IC50 = 12500 nM T20251 C9Y4EH 118720886 IC50 > 30000 nM T20251 C9SF2E 118720891 IC50 > 30000 nM T20251 CY4G7A 118720929 IC50 > 100000 nM T20251 C3BXY9 118720930 IC50 > 333000 nM T20251 CQ6U9R 118720931 IC50 > 333000 nM T20251 CYO0F9 118720932 IC50 > 100000 nM T20251 CTB1R4 118720940 IC50 = 29000 nM T20251 C9IP0Z 118720958 IC50 = 4000 nM T20251 CDN58A 118720960 IC50 > 33000 nM T20251 C70UZF 118720963 IC50 = 4000 nM T20251 C4M5WY 118720964 IC50 > 33000 nM T20251 CS73GH 118720967 IC50 = 12000 nM T20251 C30QPT 118720970 IC50 > 33000 nM T20251 CQK8L9 118720972 IC50 = 400 nM T20251 C8VYR0 118721373 IC50 = 8300 nM T20251 CE90RQ 118721374 IC50 > 100000 nM T20251 C7MN6D 118721376 IC50 = 54700 nM T20251 CPC71H 118722570 IC50 = 6900 nM T20251 CTL19H 118722571 IC50 = 6400 nM T20251 C2JGB3 118722572 IC50 = 3600 nM T20251 CKD42B 118722573 IC50 = 9400 nM T20251 C6PMQ1 118722574 IC50 > 30000 nM T20251 C3ZL5Y 118722575 IC50 = 11000 nM T20251 CR3UB2 118722576 IC50 = 5700 nM T20251 CX1W8N 118722577 IC50 > 30000 nM T20251 C49DXR 118722578 IC50 = 17000 nM T20251 CW5GK1 118722579 IC50 > 30000 nM T20251 C50GXM 118722580 IC50 > 30000 nM T20251 CEI62G 118722581 IC50 = 3600 nM T20251 C9UG3Z 118722582 IC50 = 28000 nM T20251 C5XH4V 118722583 IC50 > 30000 nM T20251 C6Q3RV 118722584 IC50 > 30000 nM T20251 CCWD82 118722585 IC50 > 30000 nM T20251 CZ0DG2 118722586 IC50 > 30000 nM T20251 CI3R9V 118722587 IC50 = 7400 nM T20251 CSWJ92 118723345 IC50 = 280 nM T20251 CJ6V0G 118723355 IC50 = 3760 nM T20251 C0J7CS 118723360 IC50 = 950 nM T20251 C4X0GY 118723362 IC50 = 2610 nM T20251 CGN4Z9 118723363 IC50 = 1540 nM T20251 CQ3JF0 118723364 IC50 = 1400 nM T20251 C0LUV6 118723826 Ki > 10000 nM T20251 CXE6I5 118723827 Ki > 10000 nM T20251 CKO8P6 118723828 Ki > 10000 nM T20251 CL6CM1 118725606 IC50 = 3000 nM T20251 CUN73P 118725613 IC50 = 1100 nM T20251 CL5K0U 118725614 IC50 = 2000 nM T20251 CXEP50 118725615 IC50 = 2300 nM T20251 C1LTN0 118725864 Ki = 7800 nM T20251 CIR0O4 118725970 Ki > 15000 nM T20251 CS6BC8 118725971 Ki > 15000 nM T20251 CDV7Z0 118725972 Ki > 15000 nM T20251 CVZ9F7 118725973 Ki > 15000 nM T20251 CX9W7R 118725974 Ki > 15000 nM T20251 C1X4CO 118725975 Ki > 15000 nM T20251 C4DVC0 118725976 Ki > 15000 nM T20251 C0SO8I 118725977 Ki > 15000 nM T20251 CXH13A 118727337 IC50 = 1060 nM T20251 C6F5AX 118727347 IC50 = 40000 nM T20251 CF39TB 118727349 IC50 = 12000 nM T20251 CBIJ20 118728075 IC50 = 394000 nM T20251 CL32ES 118728076 IC50 = 12300 nM T20251 CHP59R 118728077 IC50 = 13800 nM T20251 CZY1K8 118728078 IC50 = 7300 nM T20251 COXN68 118728079 IC50 = 24500 nM T20251 C5K6YS 118728080 IC50 > 60000 nM T20251 CQ4TP6 118728081 IC50 > 60000 nM T20251 CRNU85 118728967 IC50 > 60000 nM T20251 CJ7N4U 118728968 IC50 > 60000 nM T20251 CY0GP6 118728969 IC50 > 60000 nM T20251 C46MUV 118728970 IC50 > 60000 nM T20251 CT7AV4 118728971 IC50 > 60000 nM T20251 CGY0L7 118728972 IC50 > 60000 nM T20251 CM7DW9 118728973 IC50 > 60000 nM T20251 CL38UF 118728974 IC50 = 53300 nM T20251 CPR5B4 118728975 IC50 > 60000 nM T20251 CB0AQ3 118728976 IC50 > 60000 nM T20251 CI1L8O 118730350 IC50 = 11500 nM T20251 C6HV3B 118730351 IC50 = 12900 nM T20251 CX50MI 118730679 IC50 > 10000 nM T20251 C1WFY9 118730799 IC50 = 48400 nM T20251 CQC32W 118730800 IC50 = 7600 nM T20251 CJ0IH1 118730801 IC50 = 32600 nM T20251 CN6UX9 118730802 IC50 = 28700 nM T20251 C05UZL 118730803 IC50 = 17600 nM T20251 CTJG53 118730804 IC50 = 11500 nM T20251 CQ48NV 118730805 IC50 = 10400 nM T20251 C26OMX 118730806 IC50 = 9300 nM T20251 CB47AL 118730807 IC50 = 8400 nM T20251 CNTH27 118730808 IC50 = 8400 nM T20251 CX50CM 118730809 IC50 = 45500 nM T20251 CN26ZK 118730810 IC50 = 6800 nM T20251 C2PT0H 118730811 IC50 = 2500 nM T20251 CRUA27 118730812 IC50 = 5700 nM T20251 CKJS86 118730813 IC50 = 4600 nM T20251 CQYK51 118730814 IC50 = 3400 nM T20251 C7TJQ5 118730994 IC50 = 2100 nM T20251 CV4E7S 118730999 IC50 = 1400 nM T20251 CC2I1K 118733347 IC50 = 5200 nM T20251 C1AVK5 118733348 IC50 = 42000 nM T20251 C43XUF 118733349 IC50 > 60000 nM T20251 C7XG3O 118733350 IC50 = 14000 nM T20251 CNYV64 118733351 IC50 = 1000 nM T20251 CLI96Y 118733352 IC50 = 5900 nM T20251 C5Q2VW 118733353 IC50 = 18000 nM T20251 C5YB6G 118733354 IC50 = 44000 nM T20251 CRO7S5 118733755 IC50 > 30000 nM T20251 C2XZN0 118733756 IC50 > 30000 nM T20251 C7MRW8 118733798 IC50 = 3980 nM T20251 C6VO5G 118733806 IC50 = 2000 nM T20251 CGKD16 118734983 IC50 = 50300 nM T20251 CX7H5Q 118734985 IC50 > 30000 nM T20251 CAN90V 118735353 IC50 = 4700 nM T20251 CIY1L8 118735865 IC50 = 730 nM T20251 CLOM28 118735866 IC50 = 1750 nM T20251 C1AI3Y 118735867 IC50 = 1060 nM T20251 C87IQN 118735868 IC50 = 5900 nM T20251 CAU0F9 118735870 IC50 = 1550 nM T20251 C3ES8P 118736031 IC50 = 13.91 nM T20251 CIB75P 118736034 IC50 = 1.7 nM T20251 C8XC3Y 118736035 IC50 = 12.38 nM T20251 C7CER2 118736036 IC50 = 0.89 nM T20251 CHL4E9 118736037 IC50 = 18.37 nM T20251 C0L2KD 118736038 IC50 = 3.27 nM T20251 CWX5Y3 118736039 IC50 = 4.2 nM T20251 C7B2JW 118736040 IC50 = 1.43 nM T20251 C60KVO 118736041 IC50 = 2.49 nM T20251 CV8Y9W 118736042 IC50 = 1.6 nM T20251 CEB0Q6 118736043 IC50 = 5.22 nM T20251 CG4D0N 118736044 IC50 = 4.21 nM T20251 CMK5V7 118736045 IC50 = 0.87 nM T20251 CRW2Y1 118736046 IC50 = 1.96 nM T20251 C0U1NW 118736047 IC50 = 13.09 nM T20251 CK58FE 118736048 IC50 = 2.08 nM T20251 CBMZ68 118736049 IC50 = 6.71 nM T20251 CJ95DR 118736050 IC50 = 2.29 nM T20251 CYQ3N5 118736051 IC50 = 0.99 nM T20251 C9CE2G 118736052 IC50 = 0.39 nM T20251 CUG5T3 118736053 IC50 = 15.62 nM T20251 CYR6Z9 118736054 IC50 = 4.93 nM T20251 CA18KF 118736055 IC50 = 16.75 nM T20251 C7VT6Q 118736056 IC50 = 7.87 nM T20251 CJ4AM8 118736655 IC50 = 25700 nM T20251 C37CTY 118736656 IC50 > 60000 nM T20251 CE3JA4 118736657 IC50 = 126000 nM T20251 C64UZP 118736658 IC50 > 60000 nM T20251 C0U5IX 118736659 IC50 > 60000 nM T20251 CS5WB8 118736662 IC50 = 30500 nM T20251 CPS96F 118736663 IC50 = 11700 nM T20251 CY5SC3 118736664 IC50 = 30000 nM T20251 CE37GC 118736665 IC50 = 7300 nM T20251 CNUS74 118736667 IC50 = 2600 nM T20251 CB42EV 118736668 IC50 > 60000 nM T20251 CP9D1G 118736669 IC50 > 60000 nM T20251 CY8I6E 118736670 IC50 > 60000 nM T20251 C97CJG 118736671 IC50 > 60000 nM T20251 CJH5D7 118736673 IC50 > 60000 nM T20251 C6WQ3N 118736674 IC50 > 60000 nM T20251 CVKD56 118736675 IC50 > 60000 nM T20251 CH0R6U 118736676 IC50 > 60000 nM T20251 C8IEB7 118736677 IC50 > 60000 nM T20251 CKV91L 118736679 IC50 = 16500 nM T20251 C3IM7W 118736680 IC50 > 60000 nM T20251 C1X8EJ 118736681 IC50 > 60000 nM T20251 CG52WO 118736682 IC50 > 60000 nM T20251 C9ZQH1 118736683 IC50 = 30400 nM T20251 C06IYV 118736684 IC50 = 31600 nM T20251 CRJ38C 118736685 IC50 > 60000 nM T20251 C67WJQ 118736760 IC50 > 60000 nM T20251 C8OZ7Q 118736762 IC50 > 60000 nM T20251 C54VYM 118736763 IC50 > 60000 nM T20251 CT28OR 118736765 IC50 = 30600 nM T20251 CL38BF 118736766 IC50 > 60000 nM T20251 C3UF7B 118736767 IC50 = 28200 nM T20251 C34XVR 118736768 IC50 = 33600 nM T20251 CGR7C8 118736770 IC50 = 32 nM T20251 CJ7AU0 118736771 IC50 = 8 nM T20251 CRN35A 118736772 IC50 = 64 nM T20251 C8WD3X 118736773 IC50 = 16 nM T20251 CJ46BO 118736774 IC50 = 16 nM T20251 CB23PD 118736775 IC50 = 64 nM T20251 C9X5JA 118736776 IC50 = 64 nM T20251 C2IB6U 118736777 IC50 = 32 nM T20251 CZDH32 118736778 IC50 = 64 nM T20251 CN1XD6 118736779 IC50 = 16 nM T20251 CVN7J1 118737793 IC50 > 100000 nM T20251 CVH7A9 118737794 IC50 > 100000 nM T20251 CI53XV 118737807 IC50 > 100000 nM T20251 CFM30P 118864208 IC50 = 35000 nM T20251 C6L4OC 118864285 IC50 = 8080 nM T20251 C9DM5W 118864313 IC50 = 4750 nM T20251 CF09GY 118864337 IC50 = 135000 nM T20251 C59NDJ 118864419 IC50 = 3470 nM T20251 C8AR7P 118864437 IC50 = 9560 nM T20251 CS20BC 118864476 IC50 = 52400 nM T20251 C4D9VF 118864482 IC50 = 52600 nM T20251 CELZ36 118866105 IC50 = 6900 nM T20251 CPK47S 118868365 IC50 = 79000 nM T20251 C14DLY 118872292 IC50 > 30000 nM T20251 C5Z0XH 118911481 IC50 = 120000 nM T20251 CM59EQ 118917669 IC50 > 100000 nM T20251 C6J8YF 118917671 IC50 > 100000 nM T20251 C2RBF7 118918048 IC50 = 2340 nM T20251 CW5EM8 118934075 IC50 = 10000 nM T20251 C7VL6I 118949555 IC50 > 10000 nM T20251 CN56FH 118949563 IC50 > 10000 nM T20251 C7CPN2 118950092 IC50 > 10000 nM T20251 CWR8M4 118950147 IC50 > 10000 nM T20251 C9UHO7 118950386 IC50 > 10000 nM T20251 CI9MA2 118950452 IC50 > 10000 nM T20251 CIQ51N 118953858 IC50 = 3200 nM T20251 CHJ70O 118960212 IC50 > 10000 nM T20251 CGJ9O5 118978102 IC50 > 31622.78 nM T20251 CSWO08 119057475 IC50 = 238000 nM T20251 CPS9N3 121245322 IC50 > 63095.73 nM T20251 C8P7OW 121245346 IC50 > 31622.78 nM T20251 CFOM46 121246727 IC50 > 31622.78 nM T20251 CL5Q9G 121246911 IC50 > 31622.78 nM T20251 CAL43C 121246982 IC50 > 31622.78 nM T20251 C6XK2Y 121247103 IC50 = 25118.86 nM T20251 C5S3FA 121292609 IC50 > 10000 nM T20251 COS3K9 121304408 IC50 = 812.83 nM T20251 C9G3ZJ 121304414 IC50 = 7585.78 nM T20251 CVN57T 121304417 IC50 = 2454.71 nM T20251 C4RD9Y 121304424 IC50 = 446.68 nM T20251 CN5YP1 121304426 IC50 < 100 nM T20251 CXL97W 121304430 IC50 = 2089.3 nM T20251 CA8CY5 121304437 IC50 = 295.12 nM T20251 C1PKR0 121304441 IC50 = 2818.38 nM T20251 CWLB20 121304449 IC50 = 467.74 nM T20251 CC3MP6 121304452 IC50 = 151.36 nM T20251 CW68KD 121304458 IC50 = 2884.03 nM T20251 CVA9F4 121304464 IC50 > 10000 nM T20251 CPB58L 121304467 IC50 = 3162.28 nM T20251 CFXN81 121304470 IC50 = 251.19 nM T20251 CTCA98 121304474 IC50 < 100 nM T20251 COB2X5 121304477 IC50 = 6309.57 nM T20251 CZ0BI4 121304484 IC50 = 10000 nM T20251 CW51NQ 121304485 IC50 = 407.38 nM T20251 CX1DQ6 121304488 IC50 = 1318.26 nM T20251 CZ4D2Y 121304493 IC50 = 794.33 nM T20251 CU50JM 121304499 IC50 = 257.04 nM T20251 C7NLV2 121304500 IC50 = 2951.21 nM T20251 C18GSY 121304506 IC50 = 3630.78 nM T20251 C21MEQ 121304510 IC50 < 100 nM T20251 C7F3NO 121304514 IC50 = 691.83 nM T20251 CPNV43 121304527 IC50 = 758.58 nM T20251 CCW3A9 121304532 IC50 = 1230.27 nM T20251 CQ2UM4 121304538 IC50 = 660.69 nM T20251 CR7L0O 121304539 IC50 = 891.25 nM T20251 C2GI6S 121304542 IC50 = 933.25 nM T20251 C1AB6P 121304551 IC50 = 602.56 nM T20251 CTI6Z7 121304565 IC50 = 602.56 nM T20251 CFVP28 121304568 IC50 = 446.68 nM T20251 CO6JN7 121304569 IC50 = 120.23 nM T20251 CN05ZQ 121304574 IC50 = 7943.28 nM T20251 CU0M7B 121304590 IC50 = 190.55 nM T20251 CLZK90 121304596 IC50 = 2511.89 nM T20251 C6YLM8 121304597 IC50 = 2754.23 nM T20251 CX5MO3 121304598 IC50 = 6918.31 nM T20251 C12GJP 121304609 IC50 = 2691.53 nM T20251 C31AEQ 121304649 IC50 = 524.81 nM T20251 C2VTK5 121304654 IC50 = 2754.23 nM T20251 CSYD40 121304673 IC50 = 316.23 nM T20251 C6IB0P 121304685 IC50 > 10000 nM T20251 CU0L6A 121304697 IC50 = 4677.35 nM T20251 CNOW27 121304705 IC50 = 616.6 nM T20251 C6NA0P 121304710 IC50 = 204.17 nM T20251 CXC70Q 121304711 IC50 = 933.25 nM T20251 CE0ND7 121304744 IC50 = 223.87 nM T20251 C1MZ6T 121304754 IC50 > 10000 nM T20251 C6C9EF 121304827 IC50 > 3000 nM T20251 C5HQ4S 121304867 IC50 = 1202.26 nM T20251 C6E2VF 121305983 IC50 = 9000 nM T20251 CL8P4D 121305987 IC50 = 7400 nM T20251 CR0HG1 121313818 IC50 = 4500 nM T20251 CO97HF 121313830 IC50 = 1400 nM T20251 CCUN52 121313839 IC50 = 8000 nM T20251 C4USB9 121313840 IC50 = 5000 nM T20251 C1GPN7 121313866 IC50 > 60000 nM T20251 CML4Z3 121313870 IC50 = 4200 nM T20251 CWC64Z 121313891 IC50 = 36400 nM T20251 C37BWZ 121313899 IC50 = 45000 nM T20251 CC9A1P 121313903 IC50 = 54 nM T20251 CA5L4N 121313914 IC50 = 1500 nM T20251 C0VQ4K 121313943 IC50 = 9.5 nM T20251 CD6Z2S 121313948 IC50 = 10400 nM T20251 C5TJ0N 121313953 IC50 = 12300 nM T20251 C1H8OV 121313959 IC50 = 21900 nM T20251 CTD80X 121313965 IC50 > 60000 nM T20251 CU4CW1 121313969 IC50 = 20000 nM T20251 CFP26R 121313971 IC50 = 17200 nM T20251 CNT7G1 121313972 IC50 > 60000 nM T20251 CC1G3N 121313978 IC50 = 7600 nM T20251 C8ZC5L 121313982 IC50 = 2700 nM T20251 CR74PF 121313995 IC50 = 17600 nM T20251 CTD40H 121314002 IC50 = 4500 nM T20251 CQFC86 121314009 IC50 = 3800 nM T20251 C8I2PZ 121314020 IC50 = 9400 nM T20251 C7QK2C 121314021 IC50 = 12000 nM T20251 CJT43I 121314036 IC50 > 60000 nM T20251 C8PT6Y 121314045 IC50 = 4900 nM T20251 CH8S4J 121314048 IC50 = 4700 nM T20251 CFW68T 121314052 IC50 = 19100 nM T20251 CP13EB 121314068 IC50 = 27000 nM T20251 CAS0Y9 121315197 IC50 = 562.34 nM T20251 CRZ1V0 121315205 IC50 = 263.03 nM T20251 CV3XH6 121315206 IC50 = 1949.84 nM T20251 C4TI7P 121315244 IC50 = 200 nM T20251 CLM9E8 121315259 IC50 = 524.81 nM T20251 C7B3XN 121315293 IC50 = 3981.07 nM T20251 C9U5CV 121315295 IC50 = 134.9 nM T20251 CN39AK 121315339 IC50 = 295.12 nM T20251 C14NCL 121315356 IC50 = 144.54 nM T20251 COG90M 121315374 IC50 = 151.36 nM T20251 CEY62R 121315401 IC50 < 100 nM T20251 C0E6HD 121315586 IC50 < 100 nM T20251 CBAG84 121315634 IC50 < 100 nM T20251 C9Q2ND 121333973 IC50 > 10000 nM T20251 C5BVJ8 121351012 IC50 > 25000 nM T20251 C46DBJ 121362063 IC50 = 30000 nM T20251 COGV39 121362167 IC50 = 2600 nM T20251 CV9TX1 121399281 IC50 = 19900 nM T20251 C7IU8N 121401335 IC50 > 50000 nM T20251 C7NWK8 121401336 IC50 = 44700 nM T20251 C5RXG7 121401340 IC50 > 50000 nM T20251 CV0FH9 121401343 IC50 = 2200 nM T20251 C2WD1Q 121407246 IC50 = 5351 nM T20251 CR5HV8 121410292 IC50 = 16000 nM T20251 CVE96K 121410294 IC50 = 3300 nM T20251 CK9G7V 121410328 IC50 = 2600 nM T20251 CQ3KL4 121410329 IC50 = 1800 nM T20251 CBN62U 121410340 IC50 = 8000 nM T20251 CNF06J 121410352 IC50 = 7200 nM T20251 C91PVZ 121428416 IC50 > 30000 nM T20251 CO9SQ6 121454909 IC50 > 60000 nM T20251 CH0X4Z 121454982 IC50 > 60000 nM T20251 CT0KS4 121455652 IC50 = 54000 nM T20251 CW35TI 121455794 IC50 = 26000 nM T20251 CBL46V 121488126 IC50 > 30000 nM T20251 C3WC9Y 121488127 IC50 = 12000 nM T20251 C7X1BQ 121493987 IC50 > 60000 nM T20251 CHD26A 121596332 IC50 > 33300 nM T20251 CV06MA 122177111 IC50 > 33000 nM T20251 C2DH7M 122177112 IC50 = 29000 nM T20251 CL8GC2 122177113 IC50 = 7800 nM T20251 C0H8AW 122177723 IC50 > 30000 nM T20251 CZ1F4O 122178097 Ki > 9182 nM T20251 C2AWE9 122178128 IC50 = 1600 nM T20251 CO4Y3I 122179072 IC50 = 1170 nM T20251 C92SDF 122179073 IC50 = 22390 nM T20251 C9OQ8P 122179074 IC50 > 50100 nM T20251 C6DA3N 122179075 IC50 > 50100 nM T20251 C4RYS0 122179076 IC50 > 50100 nM T20251 C9WB6E 122179416 IC50 > 40000 nM T20251 CY6C1E 122179442 IC50 = 93560 nM T20251 C5KGV7 122179447 Ki = 290 nM T20251 CFO15B 122179448 Ki = 50 nM T20251 CJP38S 122179449 Ki = 440 nM T20251 C3FP8V 122179450 Ki = 2870 nM T20251 CQGW18 122179451 Ki = 720 nM T20251 CYW75S 122179452 IC50 = 200 nM T20251 COHA53 122179453 IC50 = 190 nM T20251 CI8H9C 122179454 IC50 = 90 nM T20251 CKZ4X8 122179455 IC50 = 340 nM T20251 CZ6U4L 122179456 IC50 = 170 nM T20251 CS12JW 122179457 IC50 = 8544 nM T20251 CEQ5M0 122179459 IC50 = 7300 nM T20251 CNP81Q 122179460 IC50 = 9600 nM T20251 C54KTN 122179461 IC50 = 3200 nM T20251 C8DLB2 122179463 IC50 = 3700 nM T20251 C56TKY 122179464 IC50 = 3200 nM T20251 C49TGA 122179465 IC50 = 4300 nM T20251 CWJ9C7 122179466 IC50 = 8500 nM T20251 CI3L7J 122179467 IC50 = 22400 nM T20251 C41LSM 122179468 IC50 = 10400 nM T20251 C4U2EY 122179469 IC50 = 1600 nM T20251 C24FUL 122179470 IC50 = 35400 nM T20251 CN2FR7 122179471 IC50 = 1100 nM T20251 CJ70OH 122179472 IC50 = 5500 nM T20251 CBAO67 122179474 IC50 = 25800 nM T20251 CQ0D2N 122179475 IC50 = 51500 nM T20251 C7FA8O 122179476 IC50 = 27900 nM T20251 CNGQ19 122179477 IC50 = 27000 nM T20251 C9CLO5 122179478 IC50 = 7700 nM T20251 CY6CB1 122179479 IC50 = 7700 nM T20251 C4MZT8 122179480 IC50 = 5500 nM T20251 CDQ37R 122179481 IC50 = 3400 nM T20251 C6FME8 122179482 IC50 = 30500 nM T20251 CO34VW 122179483 IC50 = 34500 nM T20251 C3OJS0 122180330 IC50 > 10000 nM T20251 C2WV9G 122180336 IC50 > 10000 nM T20251 CJ1AP3 122180337 IC50 = 6000 nM T20251 CBN0J2 122180338 IC50 > 10000 nM T20251 CEA80S 122180339 IC50 > 10000 nM T20251 CTG4B2 122180340 IC50 > 10000 nM T20251 CTCN25 122180342 IC50 > 10000 nM T20251 C35BFD 122180343 IC50 = 6900 nM T20251 C80QZN 122180344 IC50 = 8100 nM T20251 CDZY73 122181598 Ki = 65 nM T20251 C0AM6I 122181599 Ki = 203 nM T20251 C0HR6P 122181600 Ki = 588 nM T20251 CR5T7L 122181601 Ki = 355 nM T20251 C1TA2K 122181602 Ki = 66 nM T20251 C2YMS5 122181603 Ki = 5571 nM T20251 C7L1CN 122181604 Ki = 944 nM T20251 C15JKL 122181605 Ki = 54 nM T20251 C54PWV 122181606 Ki = 60 nM T20251 C7CRS0 122181607 Ki = 48 nM T20251 CF1A6N 122181608 Ki = 3282 nM T20251 CSF5Q3 122181609 Ki = 1196 nM T20251 CP29KL 122181610 Ki = 12 nM T20251 C3GX7Z 122181612 Ki = 0.28 nM T20251 C8IGV9 122181614 Ki = 3.4 nM T20251 CF1A8R 122181616 Ki = 17 nM T20251 C64EZY 122181618 Ki = 108 nM T20251 CK0T8W 122181620 Ki = 1179 nM T20251 C9U0MK 122181622 Ki = 63 nM T20251 CJ3MG7 122181646 Ki = 577 nM T20251 C37YWX 122181648 Ki = 122 nM T20251 C1XF3L 122181650 Ki = 176 nM T20251 C61YUM 122181652 Ki = 139 nM T20251 C29KZA 122181654 Ki = 303 nM T20251 CD9YE3 122181656 Ki = 247 nM T20251 CD6HB2 122181658 Ki = 153 nM T20251 C0TDQ1 122181660 Ki = 71 nM T20251 C8M4CH 122182156 IC50 > 100000 nM T20251 CK4A6L 122182159 IC50 = 28700 nM T20251 C1MA9K 122182829 IC50 = 49970 nM T20251 C06YKW 122182830 IC50 = 23830 nM T20251 CT6L2Q 122182831 IC50 = 21870 nM T20251 CZ45UW 122182832 IC50 = 25460 nM T20251 CA1I5D 122182833 IC50 = 22290 nM T20251 C9S2AG 122182834 IC50 = 2184 nM T20251 C2R5TF 122182835 IC50 > 60000 nM T20251 CQI46V 122182836 IC50 = 47600 nM T20251 CDQ50Z 122182837 IC50 = 21060 nM T20251 CU7NC1 122182838 IC50 = 20750 nM T20251 CGJ4S6 122182839 IC50 > 60000 nM T20251 CKR73I 122182840 IC50 = 47030 nM T20251 CE7M1W 122182841 IC50 = 17880 nM T20251 C8LIP2 122182842 IC50 > 60000 nM T20251 CWE9G8 122182843 IC50 = 24330 nM T20251 C6GTI8 122182881 IC50 = 39190 nM T20251 C0D4IR 122182882 IC50 > 60000 nM T20251 CW8L5K 122184697 IC50 > 10000 nM T20251 C2VO8E 122184845 IC50 > 40000 nM T20251 CGSF80 122184846 IC50 > 40000 nM T20251 CN4H8Q 122184847 IC50 > 40000 nM T20251 CT94PN 122184848 IC50 > 40000 nM T20251 CHW2O8 122185935 IC50 = 4300 nM T20251 C9Q6GP 122185936 IC50 = 300 nM T20251 CUR4T8 122185937 IC50 = 500 nM T20251 CZJ1F9 122185938 IC50 = 1200 nM T20251 CQ1WJ8 122185975 IC50 = 398.11 nM T20251 CKD43Z 122185976 IC50 = 501.19 nM T20251 CV6OS1 122186032 IC50 = 2400 nM T20251 C9U7CE 122186033 IC50 > 30000 nM T20251 CRN80B 122186034 IC50 > 30000 nM T20251 CR8XJ5 122186035 IC50 = 2400 nM T20251 CBNO03 122186196 IC50 = 600 nM T20251 C13DXU 122186197 IC50 > 60000 nM T20251 CZ2T0Y 122186198 IC50 = 500 nM T20251 CA0IQ6 122186199 IC50 > 30000 nM T20251 CUZ16L 122186200 IC50 = 29700 nM T20251 C64MDZ 122186201 IC50 = 39900 nM T20251 CH62CJ 122186268 IC50 > 60000 nM T20251 CEG4I0 122186270 IC50 = 2300 nM T20251 C7CLG6 122186271 IC50 = 10500 nM T20251 C59PMH 122186272 IC50 = 400 nM T20251 CV36HF 122186275 IC50 = 3500 nM T20251 CV7YJ4 122186276 IC50 = 500 nM T20251 CPWB01 122186277 IC50 = 1100 nM T20251 CKD2V7 122186847 Ki = 3300 nM T20251 CQA8B2 122187067 IC50 = 1600 nM T20251 CU4X9L 122187092 IC50 > 33000 nM T20251 CQC2K7 122187093 IC50 > 100000 nM T20251 CV3LK7 122187094 IC50 > 33000 nM T20251 CJ1I2P 122187095 IC50 = 82000 nM T20251 CWE2Q3 122187096 IC50 > 100000 nM T20251 CTHX29 122187097 IC50 > 224000 nM T20251 CAZY54 122187098 IC50 > 100000 nM T20251 C2LRE0 122187099 IC50 > 100000 nM T20251 CLD74S 122187100 IC50 > 100000 nM T20251 CZR97H 122187101 IC50 = 79000 nM T20251 C8M7AW 122187102 IC50 > 100000 nM T20251 C2EN0J 122187103 IC50 > 100000 nM T20251 C45DJR 122187104 IC50 > 100000 nM T20251 CF6U2X 122187105 IC50 > 100000 nM T20251 CGO2U9 122187106 IC50 > 100000 nM T20251 CXEH62 122187107 IC50 > 100000 nM T20251 C1X9PC 122187108 IC50 = 75000 nM T20251 C59JBF 122187726 IC50 = 4450 nM T20251 CC7W9L 122187727 IC50 = 6680 nM T20251 C2N0KO 122187728 IC50 = 4750 nM T20251 CRUK02 122187729 IC50 = 900 nM T20251 C7BF8W 122187730 IC50 = 9000 nM T20251 C9VFM5 122187799 Ki = 1900 nM T20251 C4XCP1 122187801 Ki = 8300 nM T20251 CCU2N7 122187802 Ki = 6500 nM T20251 C52XCY 122188482 IC50 = 9000 nM T20251 C2XJ7S 122188483 IC50 = 1700 nM T20251 CPW3L7 122188565 IC50 = 10000 nM T20251 CSDG34 122188566 IC50 = 5700 nM T20251 C1F2GQ 122188567 IC50 = 7700 nM T20251 C49ACM 122188568 IC50 = 4800 nM T20251 CCQ2U5 122188569 IC50 = 20000 nM T20251 CMV95H 122189010 Ki = 436 nM T20251 COAL50 122189011 Ki = 777 nM T20251 CE1P0S 122189012 Ki > 10000 nM T20251 C2KD1F 122189013 Ki = 4237 nM T20251 C3KFQ6 122189014 Ki = 1666 nM T20251 CUFN73 122190176 IC50 = 1400 nM T20251 C2H7BX 122190180 IC50 > 33000 nM T20251 CNYH67 122190199 IC50 = 900 nM T20251 CJ6FZ9 122190274 IC50 = 2400 nM T20251 CGQF31 122190276 IC50 = 700 nM T20251 CEP27O 122190278 IC50 = 6100 nM T20251 C5AFZ6 122191639 IC50 > 30000 nM T20251 C1XKA8 122191834 IC50 > 30000 nM T20251 C4NUY0 122192382 IC50 = 17000 nM T20251 C1MVP5 122192989 IC50 = 10930 nM T20251 CLHV68 122192990 IC50 = 3051 nM T20251 C4DXM3 122193184 IC50 > 13000 nM T20251 C2EHL1 122193185 IC50 > 13000 nM T20251 CFU6Z1 122193186 IC50 > 13000 nM T20251 CI74XN 122193187 IC50 > 13000 nM T20251 CJ87GI 122193188 IC50 = 32000 nM T20251 C7LU2A 122193256 IC50 = 4800 nM T20251 CJ93YN 122193259 IC50 > 33000 nM T20251 CM69QJ 122193260 IC50 = 1400 nM T20251 CQ0FE9 122193263 IC50 = 500 nM T20251 CSR2O7 122195839 IC50 > 10000 nM T20251 CP7N1K 122196372 IC50 = 850 nM T20251 C7V3BY 122196373 IC50 = 3760 nM T20251 CH7TS1 122196381 IC50 = 5980 nM T20251 C0SM9Q 122196384 IC50 = 630 nM T20251 C9BAO3 122196385 IC50 = 1010 nM T20251 CZR09C 122198706 Ki = 13000 nM T20251 CZ4U5A 122429808 IC50 > 30000 nM T20251 C0AKG9 122433571 IC50 = 17500 nM T20251 CR94XB 122442340 IC50 = 10000 nM T20251 C4CMY5 122442358 IC50 = 370 nM T20251 C4RU7S 122442363 IC50 = 82 nM T20251 CB7EI3 122442376 IC50 > 10000 nM T20251 C0E5TJ 122442379 IC50 = 1700 nM T20251 CJ12FN 122442383 IC50 > 10000 nM T20251 CMW6Q8 122442385 IC50 > 10000 nM T20251 CVO84P 122442392 IC50 > 10000 nM T20251 CO3H6P 122442396 IC50 = 200 nM T20251 C2Q4VX 122442405 IC50 > 10000 nM T20251 C6KZF3 122442410 IC50 > 10000 nM T20251 C7RD0C 122442412 IC50 = 1900 nM T20251 CC05AO 122442428 IC50 > 10000 nM T20251 CI7TA4 122442447 IC50 = 900 nM T20251 CTOZ85 122442455 IC50 > 10000 nM T20251 CHE8U1 122443093 IC50 = 500 nM T20251 CC2EZ8 122443959 IC50 > 30000 nM T20251 CH6VJ4 122453014 IC50 = 10000 nM T20251 COX7E3 122510453 IC50 > 10000 nM T20251 CME91S 122513214 Ki = 2200 nM T20251 C68PHW 122579408 IC50 > 80000 nM T20251 C2HZB8 122604308 IC50 = 20000 nM T20251 C8UL7Y 122657565 IC50 = 6380 nM T20251 C85JKN 122668190 IC50 = 1520 nM T20251 CXP73N 122678088 IC50 > 31622.78 nM T20251 C1YK2E 122678192 IC50 > 33000 nM T20251 CYJX49 123132228 IC50 > 30000 nM T20251 CK7W8B 123132907 IC50 = 3500 nM T20251 CRW0C2 123132915 IC50 = 2600 nM T20251 CKT6V0 123320121 Ki = 426 nM T20251 CBT9C4 123372252 IC50 > 40000 nM T20251 C2CHR3 123471111 IC50 = 25000 nM T20251 C0T6VF 123561371 IC50 > 20000 nM T20251 CA94XD 123818187 Ki = 13040 nM T20251 C7G6IA 123944769 IC50 > 20000 nM T20251 CT9K0V 124000588 IC50 = 8800 nM T20251 CDL2V4 124005596 IC50 > 20000 nM T20251 C5ZY7L 124114343 IC50 > 50000 nM T20251 CPO7N5 124125214 IC50 > 10000 nM T20251 C4VT3O 124127413 IC50 = 15000 nM T20251 CUO46T 124140941 IC50 = 200 nM T20251 C04VCS 124140943 IC50 = 250 nM T20251 C0UAQ6 124147818 IC50 > 30000 nM T20251 C8QAD1 124147824 IC50 = 6600 nM T20251 C9SO3J 124147915 IC50 = 980 nM T20251 CS43YV 124147927 IC50 > 30000 nM T20251 CZEC76 124147932 IC50 = 17000 nM T20251 C5B4UL 124147957 IC50 = 930 nM T20251 C1KFO8 124147973 IC50 > 30000 nM T20251 C70DOJ 124147979 IC50 > 30000 nM T20251 C2VE5C 124148108 IC50 = 7 nM T20251 C3ER2Z 124148120 IC50 = 290 nM T20251 CH7OZ3 124148123 IC50 = 1200 nM T20251 CFR2G7 124148125 IC50 = 1900 nM T20251 CEK31I 124148318 IC50 > 100000 nM T20251 C25IJY 124150428 IC50 > 30000 nM T20251 C04FYJ 124150499 IC50 > 30000 nM T20251 C5H2QB 124150512 IC50 = 4000 nM T20251 CLJ36I 124150528 IC50 > 30000 nM T20251 CE2W0X 124150540 IC50 > 30000 nM T20251 C8N5JR 124150544 IC50 > 30000 nM T20251 C9TB6E 124150550 IC50 > 30000 nM T20251 C58EUN 124150620 IC50 = 9800 nM T20251 C94XQA 124150663 IC50 = 6000 nM T20251 C6FSR3 124175917 Ki > 10000 nM T20251 C7TOU4 124175991 IC50 > 10000 nM T20251 CC1O5L 124176023 IC50 = 5300 nM T20251 C49NHK 124176024 Ki = 1100 nM T20251 C49ONG 124176026 Ki = 1400 nM T20251 CTD7Q0 124176027 Ki = 2400 nM T20251 C53AYP 124176028 Ki = 5900 nM T20251 CM56CN 124176084 Ki > 10000 nM T20251 C9RLT1 124176103 Ki = 900 nM T20251 CT6HB4 124176198 Ki = 2900 nM T20251 CL7K0C 124176200 Ki = 2900 nM T20251 CWMF80 124176201 Ki = 4900 nM T20251 CYD04K 124176232 IC50 > 10000 nM T20251 CMS9P1 124176233 IC50 > 10000 nM T20251 C7EQH8 124176242 IC50 > 10000 nM T20251 C4TQO9 124176277 IC50 > 10000 nM T20251 CGJH79 124176281 IC50 > 10000 nM T20251 CCYK63 124176287 IC50 > 10000 nM T20251 CWF7N2 124176288 IC50 > 10000 nM T20251 CK0B3W 124176291 IC50 > 10000 nM T20251 CR3I7P 124176294 IC50 > 10000 nM T20251 CNC17W 124176295 IC50 > 10000 nM T20251 CO1EA0 124176296 IC50 > 10000 nM T20251 CMG02Z 124176321 IC50 > 10000 nM T20251 C4E7VI 124176804 IC50 = 1800 nM T20251 CS9U3T 126502731 IC50 > 30000 nM T20251 C6TEJ0 126532768 IC50 = 1584.89 nM T20251 CNRI41 126533424 IC50 = 316.23 nM T20251 CG65RM 126533453 IC50 < 100 nM T20251 CRX67M 126533461 IC50 = 316.23 nM T20251 C0OPY6 126533669 IC50 = 794.33 nM T20251 CSN21X 126533798 IC50 = 125.89 nM T20251 CMHY08 126533799 IC50 = 1584.89 nM T20251 CP8W0X 126533801 IC50 = 1995.26 nM T20251 CXM45K 126533810 IC50 < 100 nM T20251 C0E7OY 126533847 IC50 = 5011.87 nM T20251 CPL62Z 126533872 IC50 = 630.96 nM T20251 C1ST0Y 126533877 IC50 = 794.33 nM T20251 CDP5C4 126533939 IC50 = 158.49 nM T20251 CX2A4N 126533957 IC50 = 2511.89 nM T20251 CIV7R0 126533969 IC50 = 3981.07 nM T20251 CC7V5Y 126533978 IC50 = 630.96 nM T20251 CI97TU 126533981 IC50 = 125.89 nM T20251 CON63X 126534012 IC50 = 251.19 nM T20251 C9G1IV 126534022 IC50 < 100 nM T20251 C9AN4B 126534041 IC50 = 158.49 nM T20251 C8JKG0 126534069 IC50 = 125.89 nM T20251 C65OJB 126534075 IC50 = 630.96 nM T20251 CA4QM3 126534084 IC50 = 1258.93 nM T20251 C3SUR8 126534086 IC50 = 199.53 nM T20251 CCX0O5 126534178 IC50 = 398.11 nM T20251 C6NU0Y 126534182 IC50 < 100 nM T20251 CNUA81 126534195 IC50 = 100 nM T20251 CIAD86 126534204 IC50 = 1258.93 nM T20251 C4R7XU 126534291 IC50 = 5011.87 nM T20251 CVBX50 126534373 IC50 = 199.53 nM T20251 CB94HO 126534441 IC50 = 2511.89 nM T20251 CSX9W5 126534443 IC50 = 794.33 nM T20251 CQ39ZD 126534462 IC50 = 199.53 nM T20251 CT75WF 126534466 IC50 = 630.96 nM T20251 C52IHK 126534498 IC50 = 398.11 nM T20251 CFA3D6 126534516 IC50 = 794.33 nM T20251 CX14VB 126534676 IC50 < 100 nM T20251 CIW18V 126534678 IC50 = 125.89 nM T20251 CJPA49 126534738 IC50 < 100 nM T20251 CG7CY3 126534740 IC50 < 100 nM T20251 CQDE96 126534746 IC50 = 1995.26 nM T20251 CIN62J 126534758 IC50 = 199.53 nM T20251 CXI58O 126534764 IC50 = 125.89 nM T20251 C0WUJ5 126534771 IC50 = 1258.93 nM T20251 CFDR90 126534824 IC50 = 158.49 nM T20251 CX9LM7 126534859 IC50 = 6309.57 nM T20251 CKN57U 126534860 IC50 < 100 nM T20251 C3YB2Z 126534863 IC50 < 100 nM T20251 CR70LT 126534933 IC50 = 1000 nM T20251 CKBT37 126534948 IC50 = 1258.93 nM T20251 C6DLR7 126534986 IC50 = 794.33 nM T20251 CR10PO 126534991 IC50 = 1258.93 nM T20251 CFT24J 126535001 IC50 = 100 nM T20251 C58EIM 126535029 IC50 < 100 nM T20251 C5HQB6 126535034 IC50 < 100 nM T20251 C9Q0VB 126535075 IC50 = 251.19 nM T20251 CIZC84 126535109 IC50 > 10000 nM T20251 CMT3Q8 126535410 IC50 = 1000 nM T20251 C5YS6F 126535470 IC50 = 501.19 nM T20251 C4TZ6I 126535517 IC50 < 100 nM T20251 CTAG09 126567264 IC50 = 3380 nM T20251 C5QT4N 126567306 IC50 = 3500 nM T20251 CCH07K 126640345 IC50 = 1750 nM T20251 CR70JL 126641909 IC50 = 8300 nM T20251 CT7M6Q 126641926 IC50 = 13200 nM T20251 CLG67Z 126641948 IC50 = 12000 nM T20251 CVAC39 126641974 IC50 = 340 nM T20251 C1ZTB7 126641995 IC50 = 15800 nM T20251 CA81IH 126642266 IC50 = 19000 nM T20251 CNJL38 126642277 IC50 = 4000 nM T20251 CIW02N 126642282 IC50 = 55000 nM T20251 CY7US6 126715366 IC50 > 33000 nM T20251 CX37RN 126715380 IC50 > 100000 nM T20251 CH6YP0 126715392 IC50 > 100000 nM T20251 C1QB5R 126715400 IC50 = 22000 nM T20251 CO2X6J 126715460 IC50 = 15000 nM T20251 C09PAE 126744799 IC50 > 10000 nM T20251 COJ60B 126744800 IC50 > 10000 nM T20251 C0FKA4 126744972 IC50 = 6300 nM T20251 CT3R2Q 126961699 IC50 = 10000 nM T20251 COF75Z 126970673 IC50 = 29000 nM T20251 CS1B2E 127020968 IC50 > 100000 nM T20251 COWC81 127025601 IC50 > 11100 nM T20251 C1HGA4 127025889 IC50 > 100000 nM T20251 CF61HD 127025890 IC50 > 11100 nM T20251 CM74CE 127025891 IC50 > 100000 nM T20251 C4D9QY 127026491 IC50 > 30000 nM T20251 CBE56W 127026514 IC50 = 2830 nM T20251 C76CNA 127027374 IC50 > 10000 nM T20251 C15EJA 127027375 IC50 = 3701 nM T20251 CK8M1R 127027397 IC50 = 7261 nM T20251 C20XMQ 127027566 IC50 = 19000 nM T20251 C1PZ5S 127027702 IC50 > 10000 nM T20251 CZVP92 127028061 IC50 = 3100 nM T20251 CZ3G8X 127028062 IC50 = 4900 nM T20251 CN32ML 127028362 IC50 = 6600 nM T20251 C8MC1I 127028408 IC50 = 9100 nM T20251 CF1HM4 127028816 IC50 = 42000 nM T20251 CJ61PC 127028946 IC50 > 10000 nM T20251 CG14NR 127029113 IC50 = 21000 nM T20251 C32VER 127029260 IC50 > 5000 nM T20251 COAM29 127029262 IC50 > 5000 nM T20251 CF1MD9 127029702 IC50 = 42000 nM T20251 CL9IY6 127029888 IC50 = 17 nM T20251 C5RFV1 127029889 IC50 = 839 nM T20251 CZDO76 127030069 IC50 > 33000 nM T20251 C8WD7N 127030070 IC50 = 26000 nM T20251 C9GHX6 127030071 IC50 = 10000 nM T20251 CZCQ82 127030226 IC50 = 158 nM T20251 C7FD0M 127030227 IC50 = 467 nM T20251 C80JUT 127030228 IC50 = 69 nM T20251 C7YE3D 127030229 IC50 = 247 nM T20251 CF0S8I 127030230 IC50 = 350 nM T20251 CT9E3O 127030231 IC50 = 634 nM T20251 C0OKZ3 127030367 IC50 = 16000 nM T20251 CEP0T2 127030368 IC50 = 14000 nM T20251 CRV2K4 127030530 IC50 = 130 nM T20251 CJI5T4 127030531 IC50 = 58 nM T20251 C1F4OY 127030547 IC50 = 1742 nM T20251 C3VFN1 127030548 IC50 = 465 nM T20251 C3TQ4U 127030549 IC50 = 1817 nM T20251 C80CHF 127030550 IC50 = 1753 nM T20251 CU5T7O 127030626 IC50 = 26000 nM T20251 CQL8J6 127030928 IC50 = 7900 nM T20251 CH93CT 127030999 IC50 = 24000 nM T20251 CMKT63 127031154 IC50 = 258 nM T20251 CR87FU 127031155 IC50 = 495 nM T20251 C1RF0I 127031156 IC50 = 316.23 nM T20251 C0A5RC 127031270 IC50 > 33000 nM T20251 CF4V0J 127031338 IC50 = 5500 nM T20251 CZ6A2D 127031339 IC50 = 11000 nM T20251 CZ6P7H 127031354 IC50 = 16000 nM T20251 C5BTJ9 127031355 IC50 = 31000 nM T20251 CB7XP0 127031356 IC50 = 24000 nM T20251 CAV6G1 127031432 IC50 = 1025 nM T20251 CMU7D8 127031454 IC50 = 144 nM T20251 C9FR7D 127031456 IC50 = 101 nM T20251 C0A3PY 127031458 IC50 = 251.19 nM T20251 CY0EJ4 127031464 IC50 = 7518 nM T20251 C4GH0Z 127031465 IC50 = 2701 nM T20251 CM89VC 127031576 IC50 > 33000 nM T20251 C98TDU 127031577 IC50 > 33000 nM T20251 C4F3QY 127031621 IC50 = 11000 nM T20251 CB7Y6D 127031622 IC50 = 4200 nM T20251 CUO4V9 127031623 IC50 = 6200 nM T20251 CVGP91 127031694 IC50 = 44900 nM T20251 C2GK1H 127031773 IC50 = 4393 nM T20251 CFG8U2 127031907 IC50 = 5300 nM T20251 CI9ZB4 127031908 IC50 = 3300 nM T20251 C3NE8G 127031909 IC50 = 7500 nM T20251 CYHK91 127032122 IC50 = 44000 nM T20251 CYAR63 127032340 IC50 = 136 nM T20251 C7XI2Z 127032341 IC50 = 2944 nM T20251 C1OE8W 127032342 IC50 = 506 nM T20251 C79DCQ 127032659 IC50 = 146 nM T20251 CDX69E 127032660 IC50 = 522 nM T20251 C2TH8G 127032662 IC50 = 87 nM T20251 CZ9LM1 127032786 IC50 = 7400 nM T20251 CYZH79 127032787 IC50 = 3000 nM T20251 C7AK5Z 127033095 IC50 = 1800 nM T20251 C3UKI0 127033096 IC50 > 33000 nM T20251 CLJ6G9 127033551 IC50 = 4026 nM T20251 C9MD2C 127033672 IC50 > 33000 nM T20251 C1YR3E 127033673 IC50 = 25000 nM T20251 C1HO7F 127033703 IC50 = 970 nM T20251 CB12AP 127033704 IC50 = 6960 nM T20251 C5ITG3 127033945 IC50 = 15000 nM T20251 C4NIU0 127034022 IC50 = 1500 nM T20251 C5NU3M 127034125 IC50 = 530 nM T20251 CLR2J7 127034153 IC50 > 30000 nM T20251 CEWM81 127034292 IC50 = 200 nM T20251 C1FBI6 127034426 IC50 = 5503 nM T20251 CLN17T 127034427 IC50 = 4895 nM T20251 CMYQ47 127034428 IC50 = 6481 nM T20251 CON9I2 127034429 IC50 = 3619 nM T20251 CKS28E 127034802 IC50 = 2650 nM T20251 CKSZ13 127035240 IC50 > 60000 nM T20251 CGV62B 127035655 IC50 = 11200 nM T20251 CZY9R4 127035656 IC50 = 4900 nM T20251 C2KC9W 127035890 IC50 = 6309.57 nM T20251 CQ9ZK4 127036284 IC50 > 12250 nM T20251 C1L7MN 127036387 IC50 = 6000 nM T20251 CZA74X 127036551 IC50 = 18200 nM T20251 CGVD97 127036552 IC50 = 3300 nM T20251 CZG07V 127036553 IC50 = 5400 nM T20251 CE7M4J 127036775 IC50 > 10000 nM T20251 CS4H9O 127037230 IC50 = 3000 nM T20251 CTG43Z 127037413 IC50 = 2500 nM T20251 C15YEC 127037414 IC50 = 1200 nM T20251 C4OZ3F 127037433 IC50 = 6500 nM T20251 CL0IJ7 127037593 IC50 = 60000 nM T20251 C7T3PJ 127037594 IC50 = 36100 nM T20251 CB41IW 127037818 IC50 = 5100 nM T20251 C7L1DB 127037832 IC50 > 30000 nM T20251 CQA4K0 127038376 IC50 = 3810.2 nM T20251 C5I1PX 127038786 EC50 = 4600 nM T20251 CLH0B9 127040096 IC50 > 31622.78 nM T20251 C60HOC 127040550 IC50 = 11000 nM T20251 C6Z9VL 127040695 Ki = 1000 nM T20251 CG74QA 127040713 Ki = 1995.26 nM T20251 C34BGK 127040715 Ki = 5011.87 nM T20251 C0J8HC 127041348 Ki = 1000 nM T20251 CG84RM 127041558 IC50 = 31000 nM T20251 CS20QX 127041559 IC50 > 60000 nM T20251 CGN34V 127041705 IC50 = 1390.1 nM T20251 CN2T3I 127041869 IC50 = 7000 nM T20251 C2BE3M 127041870 IC50 = 36000 nM T20251 CS78AZ 127041951 Ki = 3162.28 nM T20251 CU9C4S 127041952 Ki = 3162.28 nM T20251 C9HPT6 127041953 Ki = 2511.89 nM T20251 C8H1RB 127041988 IC50 = 6309.57 nM T20251 CK6S5V 127042037 EC50 = 12000 nM T20251 C31SDE 127042181 IC50 = 17000 nM T20251 CS2AP8 127042622 IC50 = 6300 nM T20251 CL40ZB 127042623 IC50 > 11100 nM T20251 CJ45OF 127042624 IC50 = 10000 nM T20251 CP9L4A 127042940 IC50 = 5600 nM T20251 CR7QK2 127043679 IC50 = 1400 nM T20251 C79PSH 127044134 IC50 = 3200 nM T20251 CO6ZX5 127045058 IC50 = 26000 nM T20251 C4SFJ8 127045059 IC50 > 30000 nM T20251 C08FHU 127045060 IC50 = 21000 nM T20251 C8FZV7 127045061 IC50 = 8600 nM T20251 C5AXB2 127045351 IC50 = 7700 nM T20251 CY8BX9 127045352 IC50 = 5700 nM T20251 CC6WS4 127045353 IC50 = 9200 nM T20251 CZ0TP1 127045361 IC50 > 30000 nM T20251 CHIN43 127046285 IC50 = 47100 nM T20251 C34REM 127046317 IC50 = 94000 nM T20251 CAG9K7 127046489 IC50 > 100000 nM T20251 CH6W2T 127046982 IC50 = 2100 nM T20251 C6DP7Y 127047275 IC50 > 100000 nM T20251 C3DVM9 127047276 IC50 > 100000 nM T20251 CJH46E 127047680 IC50 = 1400 nM T20251 CM81AR 127047922 IC50 = 48380 nM T20251 C84TQV 127048530 IC50 = 640 nM T20251 CZV7Q0 127049047 IC50 > 79432.82 nM T20251 CB54VQ 127049048 IC50 > 100000 nM T20251 CDWJ67 127049172 IC50 = 2160 nM T20251 C2TKU8 127049173 IC50 = 2680 nM T20251 CJ8SG3 127049204 IC50 = 18000 nM T20251 C7D5QM 127049475 IC50 = 17000 nM T20251 C3V9MD 127049476 IC50 = 23000 nM T20251 C9A2DS 127049825 IC50 = 1890 nM T20251 CZS1L6 127049862 IC50 = 1030 nM T20251 CZD91J 127049863 IC50 = 998 nM T20251 CUT7E8 127050751 IC50 = 1610 nM T20251 CZW39D 127050752 IC50 = 1460 nM T20251 CUVQ34 127050762 IC50 = 97000 nM T20251 C5LVW9 127050783 Ki = 217 nM T20251 CXUH85 127050784 Ki = 12 nM T20251 C4LQ7M 127050803 IC50 = 6340 nM T20251 C25HJR 127050807 IC50 = 980 nM T20251 CS6C8O 127050851 IC50 = 24000 nM T20251 C1HAU4 127050852 IC50 = 23000 nM T20251 CHVU86 127050853 IC50 = 6400 nM T20251 CWDX26 127050854 IC50 = 5200 nM T20251 C7DU0N 127050855 IC50 = 17000 nM T20251 CLX8S5 127050856 IC50 = 9300 nM T20251 C9V4EG 127051045 IC50 = 6400 nM T20251 CH46LU 127051126 IC50 > 33000 nM T20251 C39WXP 127051127 IC50 > 33000 nM T20251 C5J3KY 127051128 IC50 > 33000 nM T20251 C7E4QP 127051129 IC50 > 33000 nM T20251 C35JLQ 127051177 IC50 = 3700 nM T20251 CDJQ32 127051599 IC50 = 5400 nM T20251 C2ISZ9 127051600 IC50 = 6600 nM T20251 C61GFX 127051601 IC50 = 5200 nM T20251 CFQ2X7 127051618 IC50 = 21000 nM T20251 C4DSF7 127051619 IC50 = 27000 nM T20251 C8JMN0 127051620 IC50 = 10000 nM T20251 CTZK49 127051621 IC50 = 7200 nM T20251 C7PZM3 127051622 IC50 > 33000 nM T20251 CZO5C7 127052225 IC50 = 12000 nM T20251 COX90Y 127052226 IC50 = 22000 nM T20251 CW6BR1 127052309 Ki = 91 nM T20251 C75EAL 127052638 IC50 = 600 nM T20251 C2GY5W 127052655 IC50 > 25000 nM T20251 CBYA45 127052869 IC50 = 1450 nM T20251 C5OE2H 127053611 IC50 = 17000 nM T20251 CKIU42 127263150 IC50 = 30 nM T20251 C38WDU 129012089 IC50 = 6700 nM T20251 CJI14M 129072680 IC50 > 100000 nM T20251 COL81P 129085358 IC50 > 100000 nM T20251 CI1H4A 129085361 IC50 > 100000 nM T20251 C5M7AB 129103161 IC50 = 823.7 nM T20251 C3WIA6 129103318 IC50 = 2905.4 nM T20251 C51ZGV 129103322 IC50 = 1899.6 nM T20251 CBSW14 129116690 IC50 = 11000 nM T20251 CS6OA8 129116809 IC50 = 23000 nM T20251 CV98PG 129136448 IC50 = 23000 nM T20251 C6GC0F 129186534 IC50 = 6130 nM T20251 C8KM6N 129186554 IC50 = 2670 nM T20251 CEZT92 129186564 IC50 = 5800 nM T20251 C5KJS8 129259157 IC50 > 25000 nM T20251 CBVS14 129387808 IC50 = 4880 nM T20251 CE8TV5 129893260 IC50 > 25000 nM T20251 CIL0Z5 129907910 IC50 = 130 nM T20251 CD80OM 129909338 IC50 = 186 nM T20251 C0FM1R 130196825 IC50 = 10000 nM T20251 CYA92R 130282633 IC50 > 100000 nM T20251 CO3QE2 130282636 IC50 > 100000 nM T20251 C3M2IV 130344977 IC50 = 3200 nM T20251 CE8Q7I 130345035 IC50 = 25000 nM T20251 C01UGK 130345060 IC50 = 36000 nM T20251 CN9S7B 130345097 IC50 = 51000 nM T20251 C3CH7B 130345110 IC50 = 47000 nM T20251 C7RN8L 130345158 IC50 = 68000 nM T20251 CF20BS 130345178 IC50 = 10000 nM T20251 CMO50A 130345200 IC50 = 4600 nM T20251 C29WVS 130358344 IC50 = 29000 nM T20251 CZM13E 130358354 IC50 = 66000 nM T20251 CRSH41 130391959 IC50 > 40000 nM T20251 CDE38Y 130406760 IC50 = 7800 nM T20251 CQ2K0R 130406834 IC50 > 10000 nM T20251 C47CAY 130421765 IC50 = 19952.62 nM T20251 C84YKI 130422161 IC50 > 31622.78 nM T20251 CY14VE 130449668 IC50 = 6100 nM T20251 C7HB2T 130449692 IC50 = 9600 nM T20251 CZB60C 130449716 IC50 = 7900 nM T20251 C70SUN 130449733 IC50 > 60000 nM T20251 CZCT84 130449749 IC50 > 60000 nM T20251 C9YSZ8 130449791 IC50 = 7900 nM T20251 CK68CA 130453737 IC50 = 15000 nM T20251 CR5X1T 130453989 IC50 = 15848.93 nM T20251 CVT2U3 130454024 IC50 = 7943.28 nM T20251 CT4BY6 130454058 IC50 > 31622.78 nM T20251 CZK41V 130454091 IC50 = 31622.78 nM T20251 C2OJ3C 130454093 IC50 = 12589.25 nM T20251 CDP9S1 130470501 IC50 = 17000 nM T20251 C5U1XV 130470509 IC50 = 24000 nM T20251 CLTQ15 130470516 IC50 = 14000 nM T20251 CUO41K 130470684 IC50 = 22000 nM T20251 CPC2A7 130470749 IC50 > 27000 nM T20251 C0GD9S 131728656 IC50 = 63.1 nM T20251 C96UHE 131728658 IC50 = 128.82 nM T20251 C4Z5MQ 131839619 IC50 > 100000 nM T20251 CY3P7I 131953432 IC50 > 10000 nM T20251 CE26HW 131955087 IC50 = 500 nM T20251 CU73IM 131985420 IC50 > 31622.78 nM T20251 CQEK82 131985476 IC50 = 12589.25 nM T20251 C20ZAT 131985489 IC50 > 50118.72 nM T20251 C1IKD6 131985494 IC50 > 31622.78 nM T20251 CI6W9O 131985523 IC50 > 50118.72 nM T20251 C4A1KN 132014906 IC50 = 4500 nM T20251 CN4RF6 132019596 IC50 > 100000 nM T20251 C93UNX 132041675 IC50 = 4500 nM T20251 CX27OU 132054828 IC50 > 33000 nM T20251 C3HI8S 132141090 IC50 = 371.54 nM T20251 C5P9AV 132153537 IC50 = 223.87 nM T20251 CRH07J 132156331 IC50 = 112.2 nM T20251 CWY58Z 132185302 IC50 > 40000 nM T20251 CQL4B7 132185442 IC50 = 19530 nM T20251 CS3C8P 132471744 IC50 > 100000 nM T20251 CF73XU 132473042 IC50 > 30000 nM T20251 C5U7JM 132473043 IC50 > 30000 nM T20251 CACJ46 132489333 IC50 > 10000 nM T20251 C81YTI 132510857 IC50 > 30000 nM T20251 CX05RI 132515052 IC50 = 21527.82 nM T20251 CES7P6 132517499 IC50 = 12500 nM T20251 CJZ7Y8 132569635 IC50 > 10000 nM T20251 C0Y2TP 132585192 IC50 = 50815.94 nM T20251 CJ04HZ 132585195 IC50 > 40000 nM T20251 C6CB0I 132585204 IC50 = 23000 nM T20251 CRAG89 132609278 IC50 = 14700 nM T20251 C2F6RM 132991430 IC50 > 15000 nM T20251 C39UCD 133080605 IC50 = 2900 nM T20251 C18GQC 134128280 IC50 > 10000 nM T20251 CO1RW6 134132142 IC50 = 54570 nM T20251 C6B1EN 134133066 EC50 > 30000 nM T20251 CQ95LB 134133571 IC50 > 63095.73 nM T20251 CR8HL3 134134147 IC50 = 3467.37 nM T20251 CR6I1X 134134165 IC50 = 22000 nM T20251 CJOQ95 134134229 IC50 > 60000 nM T20251 CTJF87 134134782 IC50 > 30000 nM T20251 CB9T4J 134134906 IC50 > 10000 nM T20251 CC7OQ2 134135307 IC50 = 3400 nM T20251 CE5TV4 134135453 IC50 = 2200 nM T20251 C2OSR5 134135634 IC50 = 3290 nM T20251 C1W4DO 134135721 IC50 = 11500 nM T20251 CG5VL6 134136656 IC50 = 4660 nM T20251 CG9J7V 134136763 IC50 = 1584.89 nM T20251 CD7NA5 134138492 IC50 > 30000 nM T20251 C3W5SM 134139893 IC50 = 1000 nM T20251 CWI1J7 134140478 IC50 = 8730 nM T20251 CHG9Z5 134140686 IC50 = 39810.72 nM T20251 C6B5RW 134141023 IC50 = 5400 nM T20251 CFW7E3 134141385 IC50 = 31622.78 nM T20251 CG7CX5 134141441 IC50 = 2240 nM T20251 CW04KZ 134141466 IC50 = 2700 nM T20251 C0W3JX 134142019 IC50 > 15000 nM T20251 CF41GA 134142277 IC50 > 10000 nM T20251 CYW9L4 134142282 IC50 = 16500 nM T20251 CUZB68 134143422 IC50 = 1140 nM T20251 C2IM4X 134143913 IC50 > 63095.73 nM T20251 CAL5D8 134145302 IC50 > 10000 nM T20251 CS8D9B 134145411 IC50 = 1300 nM T20251 CQ9G7H 134145670 IC50 > 30000 nM T20251 CZXT87 134145806 IC50 = 440 nM T20251 CN35SO 134146628 IC50 > 30000 nM T20251 CX3A0W 134146922 IC50 = 10400 nM T20251 CHN1C9 134147829 IC50 = 6550 nM T20251 CFG60Q 134148895 IC50 = 9100 nM T20251 CM9ZY1 134150199 IC50 > 10000 nM T20251 CA5B2J 134150245 IC50 > 60000 nM T20251 C1PQ5T 134150412 IC50 = 19952.62 nM T20251 C0S2VH 134150637 IC50 = 3311.31 nM T20251 C6NYU2 134150754 IC50 = 9549.93 nM T20251 C4R9EG 134151006 IC50 > 15000 nM T20251 COPA84 134151189 IC50 = 4500 nM T20251 C9Z1VM 134153244 IC50 > 10000 nM T20251 C8SH1L 134154191 IC50 = 3600 nM T20251 C7H8GQ 134157229 IC50 = 7900 nM T20251 C7AFS1 134157353 IC50 > 10000 nM T20251 C80WJP 134157894 IC50 = 3310 nM T20251 CSWE45 134163712 IC50 = 11000 nM T20251 C3TW0A 134374895 IC50 > 10000 nM T20251 CVLH60 134374993 IC50 = 8000 nM T20251 C47TLY 134378796 IC50 = 20000 nM T20251 C3HC0S 134537158 IC50 = 93000 nM T20251 CQC5S9 134539527 IC50 = 1170 nM T20251 C0MV7I 134539764 IC50 = 718 nM T20251 CVR60G 134539903 IC50 = 4160 nM T20251 CLA3C8 134540034 IC50 = 3280 nM T20251 CDFE40 134540190 IC50 > 30000 nM T20251 C20HAT 134585236 IC50 = 22200 nM T20251 C6W3VL 134585536 IC50 > 30000 nM T20251 CRL3O8 134585831 IC50 = 26300 nM T20251 CJXA12 134611894 IC50 = 31622.78 nM T20251 CX0UR7 134694318 IC50 = 4500 nM T20251 CLD78B 134694953 IC50 = 8300 nM T20251 CA89MQ 134813901 IC50 > 10000 nM T20251 C45OIZ 134814269 IC50 > 33300 nM T20251 C3K5PA 134814272 IC50 = 3700 nM T20251 C13ZRU 134817449 IC50 = 3120 nM T20251 CRPH17 134817805 IC50 = 3700 nM T20251 CZB7I6 134821685 IC50 = 5460 nM T20251 CS71IF 135126189 IC50 > 30000 nM T20251 C9FUK2 135151360 IC50 > 198000 nM T20251 C0BLS7 135156185 Ki > 10000 nM T20251 CUI9X6 135156216 Ki > 10000 nM T20251 C1GY2T 135156251 EC50 > 10000 nM T20251 C2HPY7 135156445 Ki > 10000 nM T20251 CCB30F 135179035 IC50 > 198000 nM T20251 CWQ30S 135192932 IC50 = 6100 nM T20251 CQI48P 135192983 IC50 = 16000 nM T20251 CT0GQ6 135197577 IC50 > 10000 nM T20251 C87VKA 135197594 IC50 > 10000 nM T20251 CQXS07 135197635 IC50 > 10000 nM T20251 C7KXF1 135197643 IC50 > 10000 nM T20251 C14FWK 135348858 IC50 > 30000 nM T20251 CWL67T 135397764 IC50 > 50118.72 nM T20251 COK4D6 135401985 IC50 > 30000 nM T20251 C1DM3K 135401987 IC50 = 21000 nM T20251 CMH4G1 135412290 Ki > 15000 nM T20251 C47LAF 135418940 IC50 > 30000 nM T20251 CB1VD9 135426471 Ki > 15000 nM T20251 CWU95A 135445691 IC50 = 133299.95 nM T20251 C6HFC8 135450111 IC50 = 12882.5 nM T20251 C9J4ES 135503073 IC50 > 10000 nM T20251 C4PM9W 135515431 IC50 = 11481.54 nM T20251 CRM4Q8 135518358 IC50 = 28000 nM T20251 CY4MV6 135566354 IC50 > 30000 nM T20251 CYVU41 135566744 IC50 = 53500 nM T20251 CI47VJ 135566923 IC50 > 30000 nM T20251 C61CPM 135570331 IC50 = 26200 nM T20251 CCNH91 135743577 IC50 > 10000 nM T20251 CN2B3D 135747628 IC50 > 30000 nM T20251 CNI90F 135797785 Ki = 2100 nM T20251 CNQ47X 135846033 IC50 = 50.12 nM T20251 CRL10Y 135857967 IC50 > 33000 nM T20251 CI1D7K 135875806 IC50 > 10000 nM T20251 CCK5I3 135883253 IC50 = 16000 nM T20251 CBX90O 135910326 IC50 > 10000 nM T20251 C5EC2O 135910327 IC50 > 10000 nM T20251 CK8XQ2 135981707 IC50 = 1400 nM T20251 C0Y4RD 135983984 IC50 > 32000 nM T20251 C4AI7G 136030608 IC50 > 10000 nM T20251 C2HP1X 136030609 IC50 > 10000 nM T20251 CCZO92 136030610 IC50 = 870 nM T20251 CO0L9T 136056541 IC50 > 30000 nM T20251 CLIE18 136056542 IC50 = 20000 nM T20251 CN1PY3 136056548 IC50 > 30000 nM T20251 CT57ZH 136069450 IC50 = 1500 nM T20251 CFT9R3 136069453 IC50 = 20000 nM T20251 CRPQ42 136069494 IC50 = 220 nM T20251 CK8Z3V 136069521 IC50 = 1000 nM T20251 CPY1B2 136069522 IC50 = 27000 nM T20251 CX0OM4 136069523 IC50 = 7700 nM T20251 C6EU4D 136069524 IC50 = 9000 nM T20251 CQA2Z1 136069531 IC50 = 22000 nM T20251 CCH31A 136069532 IC50 = 950 nM T20251 CQ1FS4 136069563 IC50 > 60000 nM T20251 CA83VQ 136094778 Ki = 5800 nM T20251 C3ZS9L 136099767 IC50 = 6800 nM T20251 CLB4O7 136099768 IC50 = 800 nM T20251 CUG28I 136117980 Ki = 1400 nM T20251 C7GP2R 136123532 IC50 = 67000 nM T20251 C1U8TM 136160538 IC50 > 10000 nM T20251 CGX6C4 136173253 IC50 > 100000 nM T20251 CRO13K 136187001 IC50 = 400 nM T20251 CJM67G 136198642 IC50 = 1960 nM T20251 CQTB32 136205798 IC50 > 30000 nM T20251 CV8QP3 136205832 IC50 = 8100 nM T20251 CB93EM 136205833 IC50 = 13000 nM T20251 CAD80N 136245084 EC50 > 10000 nM T20251 CQ4UT7 136253018 IC50 = 2200 nM T20251 C03JRC 136253041 IC50 = 300 nM T20251 C18IDZ 136253042 IC50 = 300 nM T20251 C6ZQ3M 136253058 IC50 = 80 nM T20251 CJ32EY 136253061 IC50 = 6000 nM T20251 C5KI7Q 136264975 Ki = 1641 nM T20251 C0W8KA 136299435 IC50 = 0.95 nM T20251 C5G4ES 136299436 IC50 = 1.4 nM T20251 CN41IE 136377142 IC50 = 16000 nM T20251 CL6M4I 136377184 IC50 = 2500 nM T20251 C4OVP2 136416802 IC50 > 30000 nM T20251 C7ZCT8 136416815 IC50 > 30000 nM T20251 C94CEV 136598218 IC50 = 6000 nM T20251 C7GX9P 136598247 IC50 = 16000 nM T20251 C62TMK 136598251 IC50 = 17000 nM T20251 C5EW1N 136598257 IC50 = 270 nM T20251 CG1O5Z 136598272 IC50 = 230 nM T20251 C0JQC3 136607508 IC50 = 4500 nM T20251 CO59KS 136607554 IC50 = 14000 nM T20251 C0R2IL 136901416 IC50 > 100000 nM T20251 C91WJF 136947741 Ki = 6800 nM T20251 C4VAQ0 136966273 IC50 = 800 nM T20251 CK4CM2 137028369 IC50 > 60000 nM T20251 CKJY95 137040409 IC50 = 1000 nM T20251 CF27GZ 137062183 IC50 = 1200 nM T20251 CE1G4P 137333984 IC50 > 25000 nM T20251 C8L5PZ 137348437 IC50 = 900 nM T20251 C81LGX 137349435 IC50 > 10000 nM T20251 CW6P2I 137394489 IC50 > 30000 nM T20251 C0PL4B 137434175 IC50 = 1 nM T20251 CXZ16C 137480037 IC50 > 31622.78 nM T20251 CW8QT1 137527725 IC50 = 8100 nM T20251 CS34IR 137628304 IC50 > 25000 nM T20251 C9ACX4 137628305 IC50 > 25000 nM T20251 CP2C1J 137628306 IC50 < 10000 nM T20251 CDGB50 137628309 IC50 > 25000 nM T20251 CW8ZR6 137628310 IC50 > 25000 nM T20251 C48QKY 137628311 IC50 > 25000 nM T20251 CH5AV6 137628312 IC50 > 25000 nM T20251 CU9O3A 137628639 IC50 > 50000 nM T20251 C6B5US 137628648 IC50 > 10000 nM T20251 C3A6PQ 137628670 IC50 = 10940 nM T20251 CNXJ86 137628681 IC50 = 24600 nM T20251 CQF1N6 137631458 IC50 = 131.83 nM T20251 CFB89A 137631484 IC50 > 16000 nM T20251 C2QCA5 137631487 IC50 > 60000 nM T20251 CY6TK1 137631739 IC50 = 4900 nM T20251 C0YMI5 137631826 IC50 = 570 nM T20251 CUYN25 137631834 IC50 = 3700 nM T20251 COQ47K 137631897 IC50 = 9000 nM T20251 C62NAF 137632738 IC50 = 281.84 nM T20251 CBR0X1 137632751 IC50 = 4600 nM T20251 C5N1VU 137632947 IC50 > 30000 nM T20251 C39SCN 137632955 IC50 = 2760 nM T20251 C8JWF7 137633017 IC50 = 14700 nM T20251 CVH35W 137633042 IC50 = 3000 nM T20251 CH43XI 137633091 IC50 > 60000 nM T20251 C6VWP8 137633129 IC50 = 4190 nM T20251 C30SZG 137633174 IC50 = 19000 nM T20251 C75YBS 137633326 IC50 = 251.19 nM T20251 C05ILH 137633336 IC50 = 3200 nM T20251 CHB92M 137633815 IC50 = 4960 nM T20251 CZOD53 137633880 IC50 = 2800 nM T20251 CJLB61 137633993 IC50 = 10200 nM T20251 C8C0OE 137634027 IC50 > 30000 nM T20251 C8HPN4 137634334 IC50 > 60000 nM T20251 CU40QT 137634377 IC50 = 13700 nM T20251 C5A9LK 137634700 IC50 = 87.1 nM T20251 CLK7A3 137635011 IC50 = 13900 nM T20251 CE6ZM1 137635237 IC50 = 12000 nM T20251 CX7GA4 137635351 IC50 = 32100 nM T20251 C3XRW2 137635947 IC50 > 30000 nM T20251 CMN6T7 137636115 IC50 > 40000 nM T20251 C32TPC 137636184 IC50 = 3260 nM T20251 CGOI28 137636189 IC50 = 8230 nM T20251 C7BJY5 137636807 IC50 = 4600 nM T20251 CCE5M7 137636942 IC50 = 45300 nM T20251 C7IL4D 137637204 IC50 = 14000 nM T20251 C2B1MZ 137637375 IC50 = 33000 nM T20251 CJH2V9 137637559 IC50 > 100000 nM T20251 CC8B6T 137637727 IC50 = 398.11 nM T20251 CHI7U2 137638473 IC50 = 900 nM T20251 CC09VU 137638599 IC50 = 1900 nM T20251 C3XT2M 137638639 IC50 = 3800 nM T20251 C52GLN 137638676 IC50 = 27100 nM T20251 CXG42C 137638912 IC50 > 33000 nM T20251 CF8S5N 137639002 IC50 = 1300 nM T20251 CY6VP5 137639127 IC50 = 12100 nM T20251 CF5TI6 137639661 IC50 > 100000 nM T20251 C4DW9S 137639931 IC50 = 1900 nM T20251 C4B7UM 137640060 IC50 > 30000 nM T20251 C5KX6V 137640062 IC50 = 1400 nM T20251 CJX8N5 137640241 IC50 = 13500 nM T20251 CA0QO6 137640453 IC50 > 40000 nM T20251 CVLN62 137640626 IC50 > 30000 nM T20251 CZSJ59 137640675 IC50 > 16000 nM T20251 CX01ER 137640926 IC50 > 30000 nM T20251 C91GMY 137641491 IC50 = 49200 nM T20251 C48UDJ 137642293 IC50 = 25100 nM T20251 CY98CE 137642361 IC50 > 30000 nM T20251 C9N1IG 137642471 IC50 = 1070 nM T20251 C5OXI1 137642484 IC50 > 30000 nM T20251 CBJX42 137642666 IC50 = 400 nM T20251 CYWA72 137643103 IC50 = 3800 nM T20251 C58ISN 137643139 IC50 = 34800 nM T20251 CQ87SJ 137643211 IC50 = 15000 nM T20251 C4MN6W 137643261 IC50 = 3300 nM T20251 C9BF0V 137643369 IC50 = 6100 nM T20251 CHOI53 137643582 IC50 = 1500 nM T20251 C70XZQ 137643636 IC50 = 34010 nM T20251 CU2PD4 137643678 IC50 = 1640 nM T20251 CVP8M6 137643865 IC50 > 20000 nM T20251 CEKO63 137643918 IC50 = 18.2 nM T20251 C6FPZ5 137644016 IC50 = 5480 nM T20251 C0CI4P 137644180 IC50 = 4100 nM T20251 CO7T8B 137644182 IC50 = 3300 nM T20251 CUMA78 137644191 IC50 > 30000 nM T20251 C09FUH 137644619 IC50 = 2460 nM T20251 CHS17L 137644882 IC50 = 16200 nM T20251 CV56QL 137645221 IC50 = 16500 nM T20251 C3K5IV 137645234 IC50 = 15000 nM T20251 CC1Y6W 137645554 IC50 > 31600 nM T20251 C23IRT 137645590 IC50 = 14000 nM T20251 CY1HN6 137645732 IC50 > 30000 nM T20251 C10CBD 137646316 IC50 = 20400 nM T20251 CWG0D6 137646487 IC50 > 10000 nM T20251 CM38TQ 137646827 IC50 = 1659.59 nM T20251 CFPE40 137646880 IC50 > 30000 nM T20251 C6EKO4 137646948 IC50 = 43.65 nM T20251 C8ZB5K 137647001 IC50 > 30000 nM T20251 C4O0JE 137647028 IC50 = 10000 nM T20251 C0NWV1 137647092 IC50 = 3000 nM T20251 C4DB7J 137647113 IC50 = 29000 nM T20251 C1PSL6 137647194 IC50 > 31600 nM T20251 CG9U3X 137647321 IC50 = 6500 nM T20251 CZXR87 137647404 IC50 > 10000 nM T20251 CO5M6C 137647489 IC50 > 200000 nM T20251 C3TXN9 137647591 IC50 = 31700 nM T20251 C19CXJ 137647807 IC50 = 14000 nM T20251 C4W9ED 137647842 IC50 = 28.84 nM T20251 CCIM31 137647884 IC50 > 20000 nM T20251 CTD69B 137647980 IC50 = 1200 nM T20251 CL06NY 137648464 IC50 = 29890 nM T20251 C7UTE8 137648598 IC50 = 2900 nM T20251 CH1J9F 137648789 IC50 = 67 nM T20251 CY8NV3 137648854 IC50 = 10700 nM T20251 CO89DX 137649100 IC50 = 100 nM T20251 COLY80 137649218 IC50 > 60000 nM T20251 CUFO39 137649223 IC50 > 60000 nM T20251 C0J6GS 137649319 IC50 = 900 nM T20251 CG3X9M 137649357 IC50 = 45000 nM T20251 C7SXI2 137649457 IC50 = 11300 nM T20251 C3GP4Y 137649582 IC50 > 30000 nM T20251 C04JSE 137649716 IC50 = 10300 nM T20251 CP6F7W 137650046 IC50 > 40000 nM T20251 CV0J6S 137650114 IC50 = 19300 nM T20251 CI7F1J 137650316 IC50 = 1300 nM T20251 COH10Y 137651081 IC50 = 1800 nM T20251 COCF21 137651256 IC50 > 60000 nM T20251 CB6G5D 137651292 IC50 = 75.86 nM T20251 CANL61 137651426 IC50 > 30000 nM T20251 CVR29E 137651451 IC50 = 28400 nM T20251 CS0PU8 137651464 IC50 > 40000 nM T20251 C3Z7LM 137651481 IC50 = 35000 nM T20251 CZ89GD 137651664 IC50 > 31600 nM T20251 CGXE73 137651731 IC50 > 30000 nM T20251 CRWS26 137652032 IC50 = 5600 nM T20251 CQ96SK 137652235 IC50 = 25000 nM T20251 CLN2U7 137652270 IC50 = 83000 nM T20251 CKW9B5 137652423 IC50 > 25000 nM T20251 CINE03 137652514 IC50 = 15000 nM T20251 CZ2MT3 137652584 IC50 = 26400 nM T20251 CXR6C1 137653051 IC50 >= 100000 nM T20251 CUL85Y 137653097 IC50 = 29000 nM T20251 C65XKJ 137653127 IC50 > 60000 nM T20251 CX0YC9 137653149 IC50 = 302 nM T20251 C38FXZ 137653443 IC50 > 80000 nM T20251 CQ32NO 137653545 IC50 = 11200 nM T20251 C4AQS0 137653772 IC50 = 2900 nM T20251 CVBC79 137653856 IC50 = 2200 nM T20251 C0O5HF 137654037 IC50 > 30000 nM T20251 C46DKN 137654445 IC50 = 200 nM T20251 CU6SM3 137654538 IC50 = 12400 nM T20251 CO9SD0 137654952 IC50 = 8400 nM T20251 CV89YB 137655268 IC50 = 32600 nM T20251 C8BDX5 137655281 IC50 > 60000 nM T20251 CP5S6L 137655441 IC50 = 46000 nM T20251 CSRK73 137655508 IC50 = 5600 nM T20251 C45CQG 137655515 IC50 = 1300 nM T20251 C7HO5N 137655611 IC50 > 16000 nM T20251 C17LIA 137655641 IC50 = 6730 nM T20251 C3LG7W 137655838 IC50 = 39380 nM T20251 C1OXG8 137655944 IC50 > 10000 nM T20251 CA7B5Z 137656105 IC50 > 30000 nM T20251 CVBS03 137656215 IC50 = 13200 nM T20251 CZ4W3T 137656391 IC50 = 4800 nM T20251 CN2UE9 137656598 IC50 > 60000 nM T20251 CW1J7N 137657095 IC50 = 2500 nM T20251 CXV0H7 137657379 IC50 = 5600 nM T20251 CRT86S 137657427 IC50 = 19700 nM T20251 C6C7FX 137657428 IC50 = 2900 nM T20251 C2ME3D 137657693 IC50 = 10300 nM T20251 C1NI7Z 137657872 IC50 = 22300 nM T20251 C8YB3D 137657887 IC50 = 2450 nM T20251 C9JP7K 137657919 IC50 = 14000 nM T20251 COH35U 137657930 IC50 > 30000 nM T20251 C5ZX4W 137657934 IC50 = 390 nM T20251 CB7C5E 137657969 IC50 = 3100 nM T20251 C59BVH 137658028 IC50 = 40000 nM T20251 CF7Q6D 137658206 IC50 > 30000 nM T20251 CLT89J 137658267 IC50 = 8680 nM T20251 CLZ6F9 137658483 IC50 = 20100 nM T20251 CJY5S1 137658512 IC50 = 260 nM T20251 CA72YP 137658615 Ki > 30000 nM T20251 CD87KA 137658644 IC50 > 28700 nM T20251 C45WRB 137659034 IC50 = 75.86 nM T20251 C5PV0M 137659142 IC50 = 5000 nM T20251 C1ZH9J 137659238 IC50 = 3100 nM T20251 CF25MB 137659327 IC50 = 1000 nM T20251 C0UM2I 137659879 IC50 = 4200 nM T20251 CYI45R 137660122 IC50 = 21000 nM T20251 CR41KW 137660124 IC50 = 25000 nM T20251 C5WI8U 137660200 IC50 = 5740 nM T20251 C6GN8Z 137660334 IC50 = 6700 nM T20251 C8A3EK 137660337 IC50 = 36000 nM T20251 C1YB0M 137660460 IC50 = 870 nM T20251 CJZ1A3 137660546 IC50 > 300000 nM T20251 CIMY59 137660725 IC50 = 24200 nM T20251 CXM59Y 137660745 IC50 > 16000 nM T20251 C9QHV0 137660822 IC50 > 40000 nM T20251 C7H2LV 137660844 IC50 = 46000 nM T20251 C2KX3V 137661020 IC50 > 30000 nM T20251 CC42XJ 137661121 IC50 = 19.95 nM T20251 CL8H3R 137661393 IC50 > 10000 nM T20251 C29DMS 137661489 IC50 > 60000 nM T20251 CP4IV9 137661909 IC50 = 5150 nM T20251 CUJ2F0 137662184 IC50 = 91.2 nM T20251 CY07GS 137662191 IC50 > 30000 nM T20251 C6KYD7 137700754 IC50 > 30000 nM T20251 CM3UF7 137700779 IC50 = 4700 nM T20251 CC9K8L 137796790 IC50 = 23000 nM T20251 C3QL4O 138319676 IC50 = 32000 nM T20251 C9MNG4 138319677 IC50 = 13000 nM T20251 C7TAV3 138319685 IC50 > 100000 nM T20251 CPTE92 138319693 IC50 > 30000 nM T20251 CMP8U3 138376515 IC50 = 1900 nM T20251 CE79SV 138377584 IC50 = 45000 nM T20251 CKT7F5 138393065 Ki = 15800 nM T20251 C2QLX3 138393292 IC50 > 40000 nM T20251 CFR0X3 138454761 IC50 > 40000 nM T20251 CA3C4O 138454792 IC50 > 30000 nM T20251 CHQA31 138454800 IC50 > 40000 nM T20251 C81ILP 138471783 IC50 = 8700 nM T20251 CKDZ26 138504497 IC50 = 24000 nM T20251 CBN08I 138544609 Ki = 5400 nM T20251 CSRI06 138547901 IC50 > 40000 nM T20251 CN6M0G 138964067 IC50 > 300000 nM T20251 CV6JY5 139030528 IC50 > 50118.72 nM T20251 CI1D9F 139600335 IC50 = 28000 nM T20251 CG2NH6 139600336 IC50 = 10600 nM T20251 C0HN5J 139600337 IC50 = 3000 nM T20251 CIQ96U 141478757 IC50 = 2900 nM T20251 C9JSZ2 141529337 IC50 = 47980 nM T20251 CSE1D2 141529338 IC50 = 38920 nM T20251 C43LDR 141730928 IC50 > 30000 nM T20251 C2D9TE 141756938 IC50 = 8000 nM T20251 C53UZY 141757055 IC50 = 5300 nM T20251 C7KD9N 142533975 IC50 = 7000 nM T20251 C17XZS 142727681 IC50 > 50000 nM T20251 C3MI8P 142747294 IC50 = 4000 nM T20251 C1W8QR 145865307 IC50 > 30000 nM T20251 C9ISH6 145925685 IC50 = 4700 nM T20251 CL8VT0 145946399 IC50 > 10000 nM T20251 C54ACE 145949595 IC50 = 7943.28 nM T20251 C6P9QW 145949880 IC50 = 12589.25 nM T20251 C85SDC 145949931 IC50 = 8100 nM T20251 C9Q1TH 145950015 IC50 = 15000 nM T20251 CVK2J4 145950020 IC50 = 4700 nM T20251 CTM0N6 145950094 IC50 > 10000 nM T20251 C3ASH6 145950133 IC50 = 80 nM T20251 C91DXZ 145950201 IC50 = 25118.86 nM T20251 CAB3N0 145950456 IC50 = 2620 nM T20251 CXKB09 145950494 IC50 = 4400 nM T20251 CK64FQ 145950570 IC50 > 33000 nM T20251 C6JYA5 145950619 IC50 = 2100 nM T20251 CPE7N3 145950719 IC50 > 33000 nM T20251 CYF32C 145950953 IC50 > 30 nM T20251 CL2OR1 145950976 IC50 = 20300 nM T20251 CW6XJ2 145951187 IC50 = 14000 nM T20251 CRXJ25 145951211 IC50 > 30 nM T20251 C7Q6MF 145951374 Ki > 40000 nM T20251 CCOW60 145952011 IC50 = 27000 nM T20251 CG48IY 145952272 IC50 > 10000 nM T20251 CX2UH4 145952348 Ki > 40000 nM T20251 CVR31U 145952361 IC50 = 24000 nM T20251 CAF83G 145952396 IC50 = 1584.89 nM T20251 CCY29F 145952435 IC50 > 10000 nM T20251 CVS48W 145952572 Ki > 40000 nM T20251 CLQ6T3 145953268 IC50 = 5200 nM T20251 C60XZR 145953297 IC50 > 30 nM T20251 C2WFH6 145953847 IC50 > 33000 nM T20251 CHG09C 145953855 IC50 = 3981.07 nM T20251 CJN63M 145953914 IC50 > 10000 nM T20251 C0V8SM 145954139 IC50 > 30 nM T20251 CJ89WR 145954168 IC50 = 3207 nM T20251 CJ3P0C 145954173 IC50 = 10500 nM T20251 C25NVO 145954311 IC50 = 6309.57 nM T20251 CTRQ36 145954357 IC50 = 8900 nM T20251 CBO52Q 145954980 Ki > 40000 nM T20251 C82RDB 145955110 IC50 > 10000 nM T20251 CQ56XG 145955114 IC50 = 2700 nM T20251 CFG31P 145955509 IC50 > 10000 nM T20251 CWJ0K6 145955642 IC50 > 30000 nM T20251 C3XQ4O 145956183 IC50 = 10000 nM T20251 C4Y9RM 145956261 IC50 > 10000 nM T20251 CJ5GW3 145956273 Ki > 40000 nM T20251 C0LJB1 145956360 Ki > 40000 nM T20251 CR9DQ8 145956659 IC50 > 10000 nM T20251 CL0NH3 145956868 IC50 > 10000 nM T20251 CB74GR 145957221 IC50 > 30 nM T20251 C50ATS 145957391 IC50 = 10000 nM T20251 CLC41T 145957467 IC50 = 4.22 nM T20251 CFZJ34 145957574 IC50 = 31622.78 nM T20251 C9X4EA 145957598 IC50 = 1753 nM T20251 CILC62 145957718 IC50 = 14 nM T20251 C6R0OC 145957812 IC50 = 5700 nM T20251 CB8S9C 145957865 Ki = 28000 nM T20251 CA4C9J 145957925 IC50 = 18000 nM T20251 CTN8V5 145958082 IC50 = 8500 nM T20251 CAQ41N 145958476 IC50 = 6800 nM T20251 CQ19NA 145958506 Ki > 40000 nM T20251 C2FR5D 145958670 IC50 = 21300 nM T20251 CZK51T 145958678 Ki > 40000 nM T20251 CWT43A 145958774 IC50 = 2511.89 nM T20251 C73CBD 145959061 IC50 = 23000 nM T20251 C6T8GR 145959482 IC50 > 10000 nM T20251 CDYO54 145959735 IC50 = 27000 nM T20251 C4MDJ7 145960187 IC50 > 10000 nM T20251 C4N8XW 145960316 IC50 > 10000 nM T20251 CTVX81 145960555 IC50 > 10000 nM T20251 CZ8W1F 145960626 IC50 > 30000 nM T20251 CX3VH5 145960676 IC50 = 13000 nM T20251 C4IT2A 145960697 Ki = 12700 nM T20251 CW5AC7 145960817 Ki = 38400 nM T20251 CJ1O5H 145961103 IC50 > 30000 nM T20251 CTVR05 145961491 IC50 = 7700 nM T20251 C5ZD1H 145961500 Ki = 38200 nM T20251 CG43LE 145961709 Ki > 40000 nM T20251 CRYN14 145961777 IC50 = 25000 nM T20251 CKM9A7 145961840 IC50 > 100000 nM T20251 CTC3O8 145961901 Ki = 34000 nM T20251 CIM9O6 145961922 IC50 > 100000 nM T20251 CH3D1Z 145961966 IC50 > 10000 nM T20251 CX7FC9 145962196 Ki = 16000 nM T20251 C3FB4W 145962568 Ki = 14100 nM T20251 C3GX1E 145962661 Ki = 2200 nM T20251 C5E3RJ 145962891 IC50 = 17000 nM T20251 C6VNH3 145962956 IC50 > 30000 nM T20251 C21LTM 145963134 IC50 = 4500 nM T20251 C8CQX3 145963143 IC50 > 30000 nM T20251 CC1T5Z 145963172 IC50 > 30000 nM T20251 C0QJV2 145963337 IC50 = 4200 nM T20251 CWS86L 145963466 IC50 = 15000 nM T20251 CF7K5G 145963483 IC50 = 8600 nM T20251 CE9Q8L 145963631 IC50 = 1200 nM T20251 CW7DC0 145963634 IC50 > 10000 nM T20251 CB9S3T 145963706 IC50 > 30000 nM T20251 CW62NS 145963795 IC50 > 39810.72 nM T20251 C6NT1H 145963881 IC50 = 21000 nM T20251 CAJQ14 145964002 IC50 = 5300 nM T20251 CIAD71 145964098 IC50 > 30000 nM T20251 C6K9YI 145964252 IC50 = 350 nM T20251 CQ5XM3 145964429 IC50 = 530 nM T20251 CUQ97V 145964493 IC50 = 750 nM T20251 C9FUW4 145964611 IC50 = 2200 nM T20251 CTJI01 145964752 IC50 = 1700 nM T20251 CQZ3F7 145965198 IC50 > 30000 nM T20251 CJP34X 145965420 IC50 = 85600 nM T20251 C2WE1B 145965485 IC50 = 690 nM T20251 CSK8Y1 145965486 IC50 = 4600 nM T20251 CG5C1Y 145965772 IC50 = 5490 nM T20251 CMHZ94 145965813 IC50 = 280 nM T20251 CFP9G3 145965954 IC50 > 39810.72 nM T20251 CVF4M6 145965985 IC50 = 6800 nM T20251 CQE6K0 145966013 IC50 = 430 nM T20251 C2MS3R 145966170 IC50 = 166 nM T20251 C36CZY 145966369 IC50 = 55400 nM T20251 CJ34YW 145966384 IC50 = 1120 nM T20251 CR4AG3 145966633 IC50 = 2100 nM T20251 CS51VC 145966675 IC50 = 5700 nM T20251 C4V5QG 145966727 IC50 = 460 nM T20251 CA5NY2 145966786 IC50 = 410 nM T20251 C1WA0P 145966817 IC50 > 40000 nM T20251 CZ21YN 145967045 IC50 = 760 nM T20251 C2P3YJ 145967230 IC50 = 15000 nM T20251 CDW83M 145967332 IC50 > 40000 nM T20251 C0H5UD 145967429 IC50 = 4800 nM T20251 C3K7QC 145967522 IC50 = 1900 nM T20251 C38BZY 145967590 IC50 > 3000 nM T20251 CS9MZ3 145967758 IC50 = 16000 nM T20251 CTGF42 145967808 IC50 = 800 nM T20251 CPI9S3 145967920 IC50 = 1900 nM T20251 CZKG72 145968038 IC50 = 6309.57 nM T20251 CR36FU 145968121 IC50 = 600 nM T20251 CNR31W 145968279 IC50 = 2500 nM T20251 CNB7G5 145968344 IC50 = 400 nM T20251 C9OU8R 145968403 IC50 > 2000 nM T20251 C0XC7I 145968454 IC50 = 178 nM T20251 CQCY49 145968539 IC50 = 500 nM T20251 C7MAX3 145968702 IC50 > 30000 nM T20251 C1AW2J 145968863 IC50 = 7500 nM T20251 CQU16D 145968894 IC50 = 9500 nM T20251 CK5B1E 145969068 IC50 = 12000 nM T20251 CT4QJ0 145969110 IC50 = 2000 nM T20251 CNH7O5 145969326 IC50 = 3162.28 nM T20251 CIYJ92 145969331 IC50 = 3000 nM T20251 C3KI4V 145969352 IC50 < 1000 nM T20251 CO3QA4 145969383 IC50 = 370 nM T20251 CUI97C 145969471 IC50 > 1000 nM T20251 C6TDW9 145969499 IC50 = 800 nM T20251 C06WLJ 145969520 IC50 > 10000 nM T20251 C9TWE2 145969541 IC50 > 10000 nM T20251 CR4FH0 145969547 IC50 = 1000 nM T20251 CM60DT 145969661 IC50 = 3300 nM T20251 C7T1AN 145969666 IC50 = 940 nM T20251 CHZ7N3 145969706 IC50 = 12589.25 nM T20251 CQU2J7 145969790 IC50 = 810 nM T20251 CSUM19 145969910 IC50 = 6309.57 nM T20251 CDFU92 145969917 IC50 = 1000 nM T20251 CP0YH5 145969933 IC50 = 4800 nM T20251 C5TN8I 145969964 IC50 > 10000 nM T20251 C5J9LU 145969970 IC50 = 1000 nM T20251 CK9C0H 145970062 IC50 = 3800 nM T20251 C0WIZ5 145970221 IC50 = 3800 nM T20251 CPL40F 145970342 IC50 = 1300 nM T20251 CG9BH2 145970410 IC50 = 1000 nM T20251 CM75RU 145970450 IC50 = 1300 nM T20251 CYF0S4 145970568 IC50 < 1000 nM T20251 CMRZ53 145970708 IC50 = 410 nM T20251 C8B4IY 145970709 IC50 = 900 nM T20251 CATQ85 145970768 IC50 = 800 nM T20251 CMO6C2 145970858 IC50 = 2300 nM T20251 C5O2EA 145971149 IC50 = 900 nM T20251 CP6ET4 145971201 IC50 > 10000 nM T20251 C9R2VH 145971456 IC50 = 15000 nM T20251 C53OSI 145971666 IC50 = 18400 nM T20251 C6RS0M 145972161 IC50 = 4310 nM T20251 C64NXT 145972392 IC50 = 29.96 nM T20251 CU13IP 145972573 IC50 = 2300 nM T20251 C1KJ6X 145972784 IC50 = 25118.86 nM T20251 C8RFM3 145973261 IC50 > 33000 nM T20251 C7PTX6 145973283 IC50 = 43000 nM T20251 CS6UG1 145973762 IC50 = 211.7 nM T20251 C6OI3K 145973962 IC50 = 8100 nM T20251 CVK1O7 145974594 IC50 > 100000 nM T20251 CVM02B 145974600 IC50 > 100000 nM T20251 C6XV4Q 145974681 IC50 = 7700 nM T20251 C4UBG5 145974805 IC50 = 2200 nM T20251 CUJ43W 145975270 IC50 = 850 nM T20251 CA7DN0 145975339 IC50 = 2100 nM T20251 C9ME5T 145975612 IC50 = 2300 nM T20251 CPM02H 145975616 IC50 = 2200 nM T20251 CH30YP 145975799 IC50 > 30000 nM T20251 CY7U6W 145976048 IC50 > 39810.72 nM T20251 C9MK4Z 145976157 IC50 = 880 nM T20251 C41FLJ 145976727 IC50 = 5300 nM T20251 CKU21C 145977020 IC50 = 39900 nM T20251 CM27YI 145977049 IC50 > 100000 nM T20251 C5R7ZH 145977058 IC50 = 890 nM T20251 CT5W7C 145977076 IC50 > 30000 nM T20251 CUV49K 145977796 IC50 = 4400 nM T20251 CHD83O 145977889 IC50 = 3050 nM T20251 CWJ46S 145978007 IC50 = 8000 nM T20251 CU2A1M 145978072 IC50 > 100000 nM T20251 CUQ30C 145978119 IC50 = 1400 nM T20251 CH7G2C 145978242 IC50 = 350 nM T20251 CYH46T 145978250 IC50 = 6200 nM T20251 C4DU7J 145978279 IC50 = 380 nM T20251 CY3K9M 145978286 IC50 = 2069 nM T20251 C8UOA3 145978371 IC50 = 3.27 nM T20251 CRC96P 145978494 IC50 > 39810.72 nM T20251 CVK9J5 145978628 IC50 = 85700 nM T20251 CGW6Q5 145978668 IC50 = 16500 nM T20251 CWB3L0 145978768 IC50 = 3270 nM T20251 CJWI69 145979108 IC50 = 6371 nM T20251 COBE14 145979224 IC50 = 210 nM T20251 CQ5E8T 145980370 IC50 = 2300 nM T20251 CV85ZH 145980382 IC50 = 3160 nM T20251 CVE82W 145980394 IC50 < 300 nM T20251 CSEC23 145980764 IC50 = 55300 nM T20251 CW7I0E 145981058 IC50 > 30000 nM T20251 CGA83C 145981271 IC50 = 15000 nM T20251 CNDI08 145981275 IC50 > 10000 nM T20251 CZ70KB 145981598 IC50 > 30000 nM T20251 C0QWN2 145981606 IC50 = 3900 nM T20251 CY8IF4 145981627 IC50 > 10000 nM T20251 CG1AU0 145981699 IC50 = 16000 nM T20251 C4SKG5 145981746 IC50 = 900 nM T20251 C7AE4L 145981787 IC50 > 10000 nM T20251 CD5GI8 145982093 IC50 > 30000 nM T20251 C1BP0G 145982116 IC50 = 27500 nM T20251 CVOU09 145982242 IC50 = 50000 nM T20251 CD6IQ0 145982284 IC50 = 220 nM T20251 CZN0U6 145982478 IC50 > 10000 nM T20251 CX0P5N 145982847 IC50 = 10000 nM T20251 CL13NC 145982905 IC50 = 794.33 nM T20251 C4XQK5 145982959 IC50 = 1600 nM T20251 CF8E5K 145983040 IC50 = 1300 nM T20251 C4N5TW 145983050 IC50 = 25118.86 nM T20251 CND20U 145983060 IC50 = 3300 nM T20251 CC3SD4 145983205 IC50 = 5000 nM T20251 C1DW4U 145983928 IC50 = 7850 nM T20251 C8UI5J 145984101 IC50 = 3000 nM T20251 C7CUB1 145984146 IC50 = 26000 nM T20251 CJ70YV 145984499 IC50 = 1995.26 nM T20251 CJ8K4G 145984512 IC50 = 5600 nM T20251 C4R5NQ 145984560 IC50 = 10000 nM T20251 C4HAP0 145984727 IC50 = 2060 nM T20251 C9VMD1 145985361 IC50 = 6700 nM T20251 CI9QP2 145985779 IC50 = 6000 nM T20251 COG61P 145985793 IC50 = 3100 nM T20251 CRA6D0 145985939 IC50 = 1258.93 nM T20251 CNK1M7 145986171 IC50 = 5011.87 nM T20251 CXSB48 145986302 IC50 = 11300 nM T20251 C7J6XS 145986357 IC50 = 19952.62 nM T20251 CI9OL2 145986409 IC50 = 8000 nM T20251 C2UZ1G 145986549 IC50 = 15800 nM T20251 C9V3MF 145986593 IC50 = 12000 nM T20251 CPN29R 145986920 IC50 = 10000 nM T20251 C5R6BS 145987142 IC50 = 4600 nM T20251 CG1PV7 145987277 IC50 = 6309.57 nM T20251 CHOY46 145987281 Ki > 10000 nM T20251 C02VTZ 145987482 IC50 = 260 nM T20251 CI0PA9 145987771 IC50 = 16660 nM T20251 CZY0X1 145987861 IC50 = 2500 nM T20251 C8Q2EG 145988110 IC50 > 100000 nM T20251 CY1OF2 145988177 IC50 = 5100 nM T20251 COCV25 145988531 IC50 > 50000 nM T20251 C49EDV 145988588 IC50 = 8305 nM T20251 CUAY25 145988620 IC50 = 300 nM T20251 CGJI91 145988834 IC50 = 3800 nM T20251 CF42MQ 145988924 IC50 = 7600 nM T20251 CY3MR0 145989049 IC50 = 600 nM T20251 CEWA58 145989127 IC50 = 8000 nM T20251 CWYP01 145989394 IC50 = 950 nM T20251 CG9KC4 145989896 IC50 = 260 nM T20251 CTOL60 145990433 IC50 = 8635 nM T20251 C7GK3H 145990715 IC50 > 40000 nM T20251 CSZ4M5 145990737 IC50 > 40000 nM T20251 CMJ46R 145990794 IC50 = 7520 nM T20251 CU0K2Y 145990810 IC50 > 10000 nM T20251 CCI37B 145990833 IC50 = 1300 nM T20251 CMOY14 145991173 IC50 = 28200 nM T20251 CH5KI1 145991195 IC50 = 4600 nM T20251 C9WU5F 145991707 IC50 = 8700 nM T20251 C94VFQ 145991807 IC50 = 1340 nM T20251 C9YWM0 145991838 IC50 = 3400 nM T20251 CO49YW 145991861 IC50 = 1500 nM T20251 CR6MJ3 145992332 IC50 = 8000 nM T20251 C5LF2I 145992475 IC50 > 30000 nM T20251 C9PS8N 145993117 IC50 = 6210 nM T20251 C91EUQ 145993184 IC50 = 12100 nM T20251 CYV43P 145993203 IC50 = 210 nM T20251 C0Z6YX 145993493 IC50 = 2630 nM T20251 CE9QH0 145993537 IC50 = 16000 nM T20251 CW4O5A 145993860 IC50 > 40000 nM T20251 CN7EF3 145996526 IC50 > 40000 nM T20251 CHJ79V 145997874 IC50 > 30000 nM T20251 C3XF1S 145998078 IC50 = 30 nM T20251 CQR6C0 145998079 IC50 = 30 nM T20251 C0XEI1 145999051 IC50 > 1000 nM T20251 C6ME3G 145999062 IC50 > 1000 nM T20251 CF8Z2A 145999065 IC50 > 1000 nM T20251 CG1UY7 145999069 IC50 > 1000 nM T20251 C2KI5O 145999070 IC50 > 1000 nM T20251 CGE6S8 145999072 IC50 > 1000 nM T20251 C9XP0T 145999073 IC50 > 1000 nM T20251 CSM74D 145999085 IC50 > 1000 nM T20251 C6TK4I 145999086 IC50 > 1000 nM T20251 C9N6TA 145999163 IC50 > 1000 nM T20251 CZH5T4 145999312 IC50 > 1000 nM T20251 C4PIK7 145999315 IC50 > 1000 nM T20251 C7K0GD 145999319 IC50 > 1000 nM T20251 CY78CJ 145999744 IC50 > 1000 nM T20251 CSJ8R5 145999926 IC50 > 1000 nM T20251 CP89RK 145999927 IC50 > 1000 nM T20251 CXM20T 145999998 IC50 > 1000 nM T20251 CIL13H 145999999 IC50 > 1000 nM T20251 CW4K1Z 146000086 IC50 > 1000 nM T20251 C12WMX 146000087 IC50 > 1000 nM T20251 CAK72D 146000156 IC50 > 1000 nM T20251 C4T8EB 146000260 IC50 > 1000 nM T20251 C1ALS9 146000261 IC50 > 1000 nM T20251 CWTJ89 146000454 IC50 > 1000 nM T20251 CJ53IP 146000455 IC50 > 1000 nM T20251 CCL2Y6 146000550 IC50 > 1000 nM T20251 CR1P2S 146000752 IC50 > 1000 nM T20251 CM84OD 146001043 IC50 > 1000 nM T20251 C4HL7W 146001118 IC50 > 1000 nM T20251 C80YAQ 146001119 IC50 > 1000 nM T20251 CX8IG6 146001227 IC50 > 1000 nM T20251 C7QRP1 146001228 IC50 > 1000 nM T20251 CTYG98 146001229 IC50 > 1000 nM T20251 C2RJ1U 146176418 IC50 = 830 nM T20251 C8Z9OM 146205579 IC50 > 40000 nM T20251 CDYH19 146301731 IC50 > 30000 nM T20251 C7XPS6 146304252 IC50 > 30000 nM T20251 CFR58K 146304329 IC50 > 30000 nM T20251 C1TAC4 146499656 IC50 > 40000 nM T20251 C8P3GC 146499745 IC50 > 40000 nM T20251 C6JBU1 146538921 IC50 > 40000 nM T20251 CXG41R 146538922 IC50 > 40000 nM T20251 CSBC71 146680900 IC50 = 2400 nM T20251 C9YJZ5 147180858 IC50 = 979 nM T20251 C87WVL 147388287 IC50 = 6900 nM T20251 CB3N4D 151194558 IC50 = 180 nM T20251 C9L7IH 151773717 IC50 = 2700 nM T20251 CF4L1I 152092486 IC50 = 1530 nM T20251 CHD2X0 153404509 IC50 = 112100 nM T20251 C5LXC4 153605593 IC50 > 30000 nM T20251 CH61KN 153635907 IC50 = 160 nM T20251 C80USW 153635929 IC50 = 1520 nM T20251 CY2D5Z 153635933 IC50 = 1470 nM T20251 C2Z1JC 153635944 IC50 = 330 nM T20251 CC9LJ8 153635955 IC50 = 650 nM T20251 CV4LT9 153635960 IC50 = 1900 nM T20251 C9A5HO 153635975 IC50 = 410 nM T20251 C1SPV6 154726271 IC50 > 30000 nM T20251 CZE1S5 155126870 IC50 > 33000 nM T20251 CI6EB5 155126882 IC50 > 33000 nM T20251 CY1ZH2 155510358 IC50 = 13070 nM T20251 C2X3QO 155510360 IC50 > 30000 nM T20251 C9UF6S 155510524 IC50 = 1200 nM T20251 CYGN68 155510554 IC50 > 20000 nM T20251 CF2CU8 155510758 IC50 = 19000 nM T20251 CRD8I0 155510888 IC50 = 9410 nM T20251 C26NCB 155511048 IC50 = 4000 nM T20251 C7VS5G 155511937 IC50 = 18700 nM T20251 CXFK79 155512104 IC50 = 28200 nM T20251 CXW4J6 155512369 IC50 > 33000 nM T20251 CR1Z8A 155512529 IC50 = 2600 nM T20251 C8B0WD 155512870 IC50 > 50000 nM T20251 CVCK17 155513135 IC50 > 30000 nM T20251 C7L4TB 155513385 IC50 > 50118.72 nM T20251 CG73TZ 155513551 IC50 > 33000 nM T20251 CZEO50 155513953 IC50 = 25118.86 nM T20251 C2HPU4 155514097 IC50 = 678 nM T20251 C6M9EW 155514111 IC50 > 30000 nM T20251 CO09EN 155514507 IC50 = 4400 nM T20251 CD53LC 155514863 IC50 > 25000 nM T20251 C4JX1E 155514986 IC50 > 50118.72 nM T20251 C19KDA 155515076 IC50 = 2500 nM T20251 C86NAI 155515209 IC50 > 30000 nM T20251 C1DVH0 155515264 Ki = 1080 nM T20251 CPZ1J2 155515757 IC50 = 6400 nM T20251 CW4IZ2 155515867 IC50 > 30000 nM T20251 CCV0U2 155515900 IC50 = 5200 nM T20251 CDP7E5 155516065 IC50 > 31622.78 nM T20251 CHK09I 155516513 IC50 = 32300 nM T20251 C1OJ2X 155516584 IC50 = 8000 nM T20251 CVP8Q5 155516616 IC50 = 31120 nM T20251 CRW92X 155516645 IC50 > 30000 nM T20251 CH8YG1 155516670 Ki = 1020 nM T20251 CP1L3J 155516697 IC50 = 7100 nM T20251 C3PLC9 155516907 IC50 = 4000 nM T20251 CA3K9P 155517032 IC50 > 25000 nM T20251 C2X8HA 155517088 IC50 > 30000 nM T20251 CD9C4L 155517220 IC50 = 380 nM T20251 CY5UE9 155517299 Ki > 30000 nM T20251 CZ0RI7 155517469 IC50 = 17000 nM T20251 CYX2T8 155517511 IC50 = 26100 nM T20251 CU35GB 155517528 IC50 = 3 nM T20251 C01JPW 155517641 IC50 = 40477 nM T20251 CC2A9K 155517811 IC50 = 300 nM T20251 CXTR57 155518069 IC50 = 25900 nM T20251 CL1K2F 155518339 IC50 = 28800 nM T20251 C3XW1B 155518561 Ki = 14300 nM T20251 CRD79Z 155518589 IC50 > 25000 nM T20251 CY49NZ 155518625 IC50 > 20 nM T20251 CGCO97 155518865 IC50 = 16630 nM T20251 CVS35D 155518925 IC50 = 19000 nM T20251 CVH0P8 155519454 IC50 = 7943.28 nM T20251 CY1EN6 155519472 IC50 = 5300 nM T20251 C5KZG7 155519527 IC50 = 18000 nM T20251 C26VPM 155520046 IC50 > 10000 nM T20251 C1PJC7 155520619 IC50 > 33000 nM T20251 CKD52G 155520766 IC50 = 6060 nM T20251 CM0IC7 155521232 IC50 = 7943.28 nM T20251 C76JKY 155521282 Ki > 30000 nM T20251 CY2CK4 155521688 IC50 = 7500 nM T20251 C1M6KY 155521903 IC50 = 400 nM T20251 CQ06BH 155521919 IC50 = 38000 nM T20251 CZ8FN1 155522016 IC50 = 17270 nM T20251 CX41RI 155522177 IC50 = 21100 nM T20251 CGQ1X0 155522363 IC50 > 10000 nM T20251 C0ZXV4 155522886 IC50 > 25000 nM T20251 CAL9M0 155523067 IC50 > 50118.72 nM T20251 CAGO28 155523111 IC50 = 2110 nM T20251 CM1BV9 155523387 Ki > 60000 nM T20251 CH06BN 155523388 Ki = 820 nM T20251 CES5L2 155523448 IC50 > 10000 nM T20251 C37RVF 155523599 IC50 = 1500 nM T20251 C2LO4Y 155523731 IC50 > 25000 nM T20251 C15BIV 155523740 IC50 = 4200 nM T20251 C38OCA 155524170 IC50 = 2920 nM T20251 CVA8H7 155524476 IC50 > 30000 nM T20251 CLMK45 155524544 IC50 > 40000 nM T20251 C2EHI7 155524928 IC50 = 15848.93 nM T20251 CG71WI 155525128 IC50 > 25000 nM T20251 C94NTW 155525132 Ki = 9200 nM T20251 CMY98L 155525177 IC50 = 5600 nM T20251 C7E3UM 155525341 IC50 > 40000 nM T20251 CY7EM6 155525492 IC50 = 5 nM T20251 CZW45D 155525803 IC50 > 63095.73 nM T20251 C24PLM 155525923 IC50 = 553 nM T20251 CX59UT 155526046 IC50 = 1.1 nM T20251 CSI0N2 155526143 IC50 > 10000 nM T20251 C3W1DA 155526172 IC50 > 30000 nM T20251 CIR3K1 155526251 IC50 > 50118.72 nM T20251 CS05UF 155526423 IC50 > 10000 nM T20251 C17HOP 155526864 IC50 = 35500 nM T20251 CQ4XA9 155527433 IC50 > 20000 nM T20251 CL8Z3K 155527451 IC50 > 50118.72 nM T20251 C04OAY 155527550 IC50 = 50100 nM T20251 CT4B0F 155527719 Ki = 20050 nM T20251 C0DZ9X 155527985 IC50 = 7943.28 nM T20251 C05QTC 155528035 IC50 > 25000 nM T20251 CS0ER5 155528109 IC50 = 6100 nM T20251 CT1JB7 155528212 Ki = 3750 nM T20251 CHR60D 155528366 Ki = 10700 nM T20251 CN7I6O 155528434 Ki = 10750 nM T20251 CRGO31 155528777 IC50 = 17100 nM T20251 C5H9NQ 155529107 IC50 > 10000 nM T20251 C5QA2B 155529241 IC50 > 25000 nM T20251 C9L6OC 155529247 IC50 > 30000 nM T20251 C9U8FN 155529326 Ki > 30000 nM T20251 CW5TM8 155529670 IC50 > 31622.78 nM T20251 C8UM7E 155530060 IC50 > 10000 nM T20251 CFRQ41 155530069 IC50 = 32850 nM T20251 C4F7WU 155530183 IC50 = 8780 nM T20251 CBOJ48 155530271 IC50 > 50118.72 nM T20251 CQ6F7O 155530369 IC50 > 25000 nM T20251 C2WPD6 155530588 IC50 = 11000 nM T20251 C4L7ZO 155530653 Ki = 4100 nM T20251 CYH2Z6 155530878 IC50 = 14000 nM T20251 CCGZ20 155530937 IC50 > 32000 nM T20251 C5N7PS 155530991 IC50 = 2360 nM T20251 C86HGK 155531857 IC50 = 22000 nM T20251 CY59IV 155531989 IC50 = 1.4 nM T20251 CW14TB 155532044 IC50 = 1480 nM T20251 CQU09F 155532106 IC50 = 10000 nM T20251 CFL61W 155532250 IC50 > 10000 nM T20251 CZF0X4 155532360 IC50 > 10000 nM T20251 C7UBH8 155532385 Ki = 20230 nM T20251 CWEZ83 155532537 IC50 > 10000 nM T20251 C8IP7E 155532982 IC50 > 20000 nM T20251 CFR56S 155533031 IC50 > 50118.72 nM T20251 C5TFA7 155533222 IC50 > 10000 nM T20251 CAT9V1 155533370 IC50 > 30000 nM T20251 C6R8JM 155533521 IC50 > 50118.72 nM T20251 CZ3DW6 155533821 IC50 > 30000 nM T20251 CF2MD7 155533927 Ki = 24800 nM T20251 CGH63O 155534464 IC50 = 5400 nM T20251 CL7U8D 155534608 IC50 = 3 nM T20251 C82LDF 155534740 IC50 > 50118.72 nM T20251 C63HSA 155534748 IC50 > 30000 nM T20251 CVBC47 155535120 IC50 = 12000 nM T20251 C71YMQ 155535169 IC50 < 100 nM T20251 CNA92P 155535177 IC50 = 30000 nM T20251 CX7PM4 155535638 IC50 > 12589.25 nM T20251 CC5HJ6 155535796 IC50 = 18900 nM T20251 CHOC87 155535920 IC50 = 40000 nM T20251 C9JD7A 155535968 IC50 = 39810.72 nM T20251 C3F8NR 155536006 IC50 > 31622.78 nM T20251 C0BH6W 155536009 IC50 > 25000 nM T20251 CN07PE 155536057 IC50 > 30000 nM T20251 CDL9R5 155536374 IC50 = 5248.07 nM T20251 C52GJS 155536419 IC50 = 1500 nM T20251 CRI0X6 155536978 IC50 = 3200 nM T20251 CG6P2Z 155537026 IC50 = 80000 nM T20251 CY32TQ 155537053 IC50 = 8100 nM T20251 C8YO9Q 155537362 IC50 = 4 nM T20251 CY3S0M 155537382 IC50 = 14000 nM T20251 CL53AK 155537567 IC50 = 21700 nM T20251 CM3PB2 155537682 IC50 > 25000 nM T20251 CA0T9E 155537745 IC50 = 8450 nM T20251 CG8I5F 155538033 IC50 > 33000 nM T20251 C2APW9 155538169 IC50 = 32000 nM T20251 C6KX1G 155538348 IC50 = 6300 nM T20251 C4OEL6 155538351 IC50 = 5011.87 nM T20251 CUS3I9 155538644 IC50 > 25000 nM T20251 C8QX7D 155538795 Ki = 1200 nM T20251 CKNZ09 155539203 IC50 = 2900 nM T20251 CF6E1H 155539416 IC50 = 4740 nM T20251 CXV14T 155539760 IC50 = 2100 nM T20251 CCG68S 155539794 IC50 > 30000 nM T20251 C5Y4UG 155540068 IC50 = 2500 nM T20251 CK1G0I 155540170 IC50 = 4100 nM T20251 CD6J8H 155540340 IC50 = 2700 nM T20251 CDQF20 155540443 IC50 > 30000 nM T20251 CW2V3F 155540455 IC50 = 3000 nM T20251 CSMI71 155540479 Ki = 8200 nM T20251 CP2NY0 155540484 IC50 > 100000 nM T20251 C7LIO1 155540498 IC50 = 590 nM T20251 CFW15C 155540816 IC50 = 8540 nM T20251 C8WRH2 155540919 IC50 = 6400 nM T20251 CH6ND7 155541175 IC50 = 356180 nM T20251 C2IJL1 155541368 IC50 > 30000 nM T20251 CWQ7F0 155541490 IC50 = 5 nM T20251 CP2K9D 155541549 IC50 = 4400 nM T20251 C9SIN5 155541564 IC50 = 22000 nM T20251 C13HGT 155541849 IC50 = 2100 nM T20251 CQI12H 155541951 Ki = 2940 nM T20251 CL18DI 155542104 IC50 = 2200 nM T20251 C8PS6H 155542274 IC50 = 67800 nM T20251 C5T9KE 155542416 IC50 > 30000 nM T20251 CGKM58 155542422 IC50 = 17600 nM T20251 C2ZNB4 155542480 IC50 = 3900 nM T20251 CIPG54 155542639 IC50 = 3600 nM T20251 CWO01S 155542792 IC50 = 1700 nM T20251 CY8PB1 155542894 IC50 = 4000 nM T20251 CVNR95 155542898 IC50 > 30000 nM T20251 CDZ78J 155542932 IC50 = 6310 nM T20251 CU6H9N 155543153 IC50 > 10000 nM T20251 CKIJ48 155543371 IC50 = 360 nM T20251 C1FG3H 155543475 IC50 = 4500 nM T20251 CG7D9R 155543873 IC50 = 3300 nM T20251 CL9Z6H 155543895 IC50 = 7560 nM T20251 CF1AJ2 155544000 IC50 = 25118.86 nM T20251 CST86Y 155544326 Ki = 6540 nM T20251 CD9KW4 155544699 Ki = 18980 nM T20251 C8WGH1 155544876 IC50 = 12589.25 nM T20251 C7SQX2 155544997 IC50 = 1100 nM T20251 CURJ73 155545015 IC50 = 11000 nM T20251 C4I9LA 155545020 IC50 = 17900 nM T20251 CND38C 155545031 IC50 > 100000 nM T20251 CPB87M 155545130 IC50 = 1.7 nM T20251 C9H1RS 155545131 IC50 = 3600 nM T20251 CK4OU8 155545400 Ki = 9800 nM T20251 C9BVD8 155545737 IC50 > 50000 nM T20251 C8YG3O 155545771 IC50 > 10000 nM T20251 C2E5BY 155545899 IC50 > 30000 nM T20251 CB62FS 155546028 IC50 = 5400 nM T20251 CUI35S 155546230 IC50 = 13200 nM T20251 C6KXY5 155546286 IC50 = 2300 nM T20251 CPK82D 155546294 IC50 = 13000 nM T20251 CQSI68 155546312 IC50 > 10000 nM T20251 CD2PX1 155546796 IC50 = 9900 nM T20251 CI92YC 155546800 Ki = 12120 nM T20251 C7LZ3W 155546850 IC50 = 39810.72 nM T20251 C0VY9U 155547183 Ki = 5900 nM T20251 CH94MI 155547266 IC50 = 5500 nM T20251 CRN8Z6 155547317 IC50 > 31622.78 nM T20251 CQ6D2C 155547369 IC50 > 40000 nM T20251 CC83QJ 155547453 IC50 > 10 nM T20251 CU2QO9 155547462 IC50 = 8900 nM T20251 CQ62MW 155547536 IC50 = 450 nM T20251 CZ30SI 155547634 IC50 = 6309.57 nM T20251 CY6F3D 155547951 IC50 = 1600 nM T20251 CK3B4X 155548125 IC50 = 5900 nM T20251 CG8FO4 155548512 IC50 = 1100 nM T20251 CFD4W6 155548620 IC50 > 10000 nM T20251 C14SPW 155548636 IC50 = 8950 nM T20251 CRY3A2 155548898 IC50 > 30000 nM T20251 CNX8L6 155549162 Ki = 4100 nM T20251 CTQ9Y4 155549436 IC50 > 10000 nM T20251 CJD38X 155549583 IC50 = 10000 nM T20251 C0DHX7 155550192 IC50 = 1071.52 nM T20251 C8JI1D 155550286 IC50 = 1200 nM T20251 CAJ57R 155550406 IC50 = 2000 nM T20251 CEDN41 155550408 IC50 = 3 nM T20251 CR8DO6 155550599 IC50 = 830 nM T20251 C29BAV 155550731 IC50 = 1750 nM T20251 CWC8X9 155550748 IC50 > 30000 nM T20251 CHDG36 155550819 IC50 > 25000 nM T20251 CA5G2T 155551013 IC50 = 15300 nM T20251 CN9LP5 155551221 IC50 = 15000 nM T20251 CB73CQ 155551312 IC50 = 4 nM T20251 CZ7K0T 155551653 IC50 > 10000 nM T20251 C5LTO0 155551695 IC50 = 620 nM T20251 CK5F8L 155551725 IC50 > 10000 nM T20251 C5T3VG 155551984 IC50 = 13000 nM T20251 CJL9K4 155552042 IC50 = 1900 nM T20251 C26SHF 155552468 IC50 > 10000 nM T20251 CK52WB 155552587 IC50 = 1260 nM T20251 CGV1M3 155552611 IC50 = 3500 nM T20251 C1DV5G 155552667 IC50 = 21100 nM T20251 CX6QO1 155552713 IC50 = 670 nM T20251 CEN80B 155552714 IC50 = 1600 nM T20251 C2ZNL8 155552880 IC50 = 4300 nM T20251 C2QPM5 155553335 IC50 = 500 nM T20251 CN1B6E 155553350 IC50 = 1408 nM T20251 CUH7R2 155553391 IC50 > 10000 nM T20251 CORH39 155553574 IC50 > 20000 nM T20251 CT9S6V 155553775 IC50 > 10000 nM T20251 C09TOV 155553799 IC50 = 3600 nM T20251 CH18PL 155553803 IC50 = 19700 nM T20251 C7JCS2 155553955 IC50 > 25000 nM T20251 CRI95M 155554023 IC50 > 50000 nM T20251 CHP3R7 155554099 IC50 = 2100 nM T20251 C0I4KF 155555078 IC50 = 18000 nM T20251 CF78YP 155555080 IC50 > 30000 nM T20251 CGJO65 155555092 IC50 = 10600 nM T20251 CS8C4B 155555411 IC50 = 2800 nM T20251 C7TAB2 155555536 IC50 = 3100 nM T20251 C8Q2FG 155555556 IC50 > 30000 nM T20251 C76IMR 155555589 IC50 = 3500 nM T20251 C09FGY 155555863 IC50 > 25000 nM T20251 COK95C 155555928 IC50 > 12589.25 nM T20251 CRA05Z 155555980 IC50 > 12589.25 nM T20251 CFRD75 155555996 Ki > 40000 nM T20251 CIK75H 155556042 IC50 > 25000 nM T20251 C3TZ1X 155556063 IC50 = 9600 nM T20251 C8PI6V 155556175 Ki = 3560 nM T20251 CL8K4E 155556216 IC50 > 50000 nM T20251 CG80ZH 155556340 IC50 = 13300 nM T20251 C3WT2Q 155556441 IC50 > 30000 nM T20251 C7AZ5J 155556578 IC50 > 50118.72 nM T20251 CIY5U0 155556737 IC50 = 19952.62 nM T20251 C4AG5W 155557133 IC50 > 10000 nM T20251 CHVI34 155557396 IC50 = 2000 nM T20251 CK52DB 155557515 IC50 = 1400 nM T20251 CEX1O2 155557657 IC50 = 2350 nM T20251 C0T6WM 155558045 Ki > 30000 nM T20251 C2A1ZD 155558144 IC50 > 10000 nM T20251 CXD56L 155558183 IC50 > 10000 nM T20251 CR41JN 155558349 Ki = 5700 nM T20251 C92NTS 155558433 IC50 = 2500 nM T20251 CP31BL 155558617 IC50 > 1000 nM T20251 C4HPK2 155558743 IC50 > 25000 nM T20251 C9D1UW 155558867 IC50 = 7840 nM T20251 C4D1AF 155559052 IC50 = 18200 nM T20251 CJ82WQ 155559138 IC50 > 100000 nM T20251 CM0UH7 155559265 IC50 > 20 nM T20251 CKZT21 155559364 IC50 > 33000 nM T20251 C2AGR5 155559542 IC50 = 240 nM T20251 CTI7O1 155559782 IC50 = 10000 nM T20251 CKT84D 155559905 IC50 = 5200 nM T20251 CEF9N6 155560028 IC50 < 10000 nM T20251 C1U4ZL 155560181 IC50 = 280 nM T20251 CF4LM6 155560880 IC50 > 25000 nM T20251 CW3RA2 155561008 IC50 = 2500 nM T20251 CZ4BY2 155561096 Ki > 25000 nM T20251 CLO3B1 155561152 IC50 = 12000 nM T20251 CM7ZG9 155561160 IC50 > 25000 nM T20251 C9UYA8 155561280 IC50 = 5100 nM T20251 COSE65 155561444 IC50 = 10000 nM T20251 CM9L3Z 155561503 IC50 > 25000 nM T20251 C9HIU5 155561551 IC50 > 25000 nM T20251 CH9UY6 155562079 IC50 = 10000 nM T20251 C6T2RV 155562253 IC50 < 10000 nM T20251 CP52DQ 155562348 IC50 = 760 nM T20251 CS3T7F 155562863 IC50 = 2400 nM T20251 CWM03V 155563050 IC50 > 30000 nM T20251 CM23AF 155563334 IC50 > 10000 nM T20251 C85CNT 155563518 IC50 = 600 nM T20251 CAN0G3 155563660 IC50 = 1183 nM T20251 CG9QR6 155563968 IC50 = 680 nM T20251 CWOE21 155564042 IC50 > 30000 nM T20251 CFT46O 155564074 IC50 = 15000 nM T20251 CZ6TP2 155564129 IC50 = 300 nM T20251 CU7O1C 155564384 Ki = 18100 nM T20251 CZR6W0 155564401 IC50 = 1700 nM T20251 CMK03D 155564568 IC50 > 25000 nM T20251 CC5FE7 155564581 IC50 > 30000 nM T20251 CB7SJ5 155564720 IC50 = 570 nM T20251 CMR8A9 155565213 IC50 > 10000 nM T20251 CWK95R 155565459 IC50 = 17000 nM T20251 CEO89S 155565478 IC50 = 2600 nM T20251 CL63KT 155565570 IC50 = 904350 nM T20251 CJL8Y5 155565696 Ki > 30000 nM T20251 C43CBF 155566090 IC50 = 6 nM T20251 CX52IW 155566155 IC50 = 7830 nM T20251 C7WTF8 155566556 IC50 = 1700 nM T20251 C26IRL 155566625 IC50 = 1500 nM T20251 CTVY40 155566771 IC50 = 4500 nM T20251 CC2Q9P 155566780 IC50 = 109010 nM T20251 CUIS06 155566980 IC50 = 5800 nM T20251 CXKI62 155567017 IC50 = 2300 nM T20251 C8HR4Q 155567029 IC50 = 2030 nM T20251 C5YX9V 155567261 IC50 = 20380 nM T20251 C37BGO 155567311 IC50 > 30000 nM T20251 C9KQW3 155567372 IC50 = 1900 nM T20251 C08ZCY 155567532 IC50 > 30000 nM T20251 C7KPT9 155567536 IC50 = 3100 nM T20251 CU34OH 155567589 IC50 > 10000 nM T20251 C16AQH 155567592 IC50 > 30000 nM T20251 CB19FR 155567818 IC50 > 40000 nM T20251 CD5FO3 155567866 IC50 > 50118.72 nM T20251 CK9N0Z 155567885 Ki > 10000 nM T20251 CS9GW7 155568268 IC50 = 11000 nM T20251 C9ZR8N 155568412 IC50 = 25100 nM T20251 CR5HK7 155568706 IC50 = 9400 nM T20251 C8INK5 155568740 IC50 = 11000 nM T20251 CUT84A 155568798 IC50 = 1000 nM T20251 C1S8ZB 155568922 IC50 = 2300 nM T20251 CSC8Q5 155569142 IC50 = 9500 nM T20251 CBJ5F8 155569464 IC50 = 2200 nM T20251 CP9TR0 10324985 Ki > 10000 nM T20251 CB0I4L 24884859 IC50 = 8111.11 nM T20251 C7Y0EQ 24885255 IC50 = 9500 nM T20251 CYV2S9 24885661 IC50 = 750 nM T20251 C5Z2KD 24886136 IC50 = 571.43 nM T20251 CS5N4V 24886137 IC50 = 296.7 nM T20251 CP2O0E 24886138 IC50 = 2555.56 nM T20251 CZO3R2 24886366 IC50 = 7714.29 nM T20251 C90ROZ 24886368 IC50 = 1109.59 nM T20251 C7BYA1 44254046 IC50 = 2000 nM T20251 C65JLI 44254219 IC50 = 1166.67 nM T20251 D00AWM 9826520 IC50 = 1170 nM T20251 D00CCV 11669239 Ki = 2200 nM T20251 D00FAY 13007806 IC50 = 1500 nM T20251 D00NCL 46836562 IC50 = 28000 nM T20251 D00TGC 56951318 Ki > 15000 nM T20251 D00UIN 11739248 IC50 = 1000 nM T20251 D00WKK 11710246 IC50 > 60000 nM T20251 D01ABR 44414723 IC50 = 5840 nM T20251 D01BWV 9802572 IC50 = 150 nM T20251 D01FFX 24691160 Ki = 3800 nM T20251 D01GPC 53235534 IC50 = 19000 nM T20251 D01IWD 159502 IC50 = 5888.44 nM T20251 D01JYY 11323940 Ki = 7000 nM T20251 D01MCD 25059294 IC50 = 120 nM T20251 D01PIU 44297094 IC50 = 3467368.5 nM T20251 D01PYU 9821248 Ki = 530 nM T20251 D02BPT 942 IC50 = 245470.89 nM T20251 D02DCM 44230874 IC50 = 9000 nM T20251 D02EIB 25129433 IC50 = 643 nM T20251 D02FQG 54579974 IC50 = 8240 nM T20251 D02NMN 23634102 IC50 = 31000 nM T20251 D02QJW 2798 IC50 = 12.59 nM T20251 D02TPY 25025860 IC50 = 1200 nM T20251 D02TSN 46244454 IC50 = 50000 nM T20251 D02WWM 175064 IC50 = 2.188 nM T20251 D03BQV 3033806 IC50 > 10000 nM T20251 D03NRJ 10871642 Ki = 2500 nM T20251 D03PIP 11568942 Ki = 2400 nM T20251 D03PSY 44542667 IC50 = 10 nM T20251 D03RBD 49765077 IC50 = 0.26 nM T20251 D03WAE 1301094 Ki = 4.8 nM T20251 D03XKL 11641429 Ki = 300 nM T20251 D04ALU 3076 IC50 = 17378.01 nM T20251 D04SAO 9799518 IC50 > 100000 nM T20251 D04TPA 72163809 IC50 = 21000 nM T20251 D04TWX 9794475 Ki > 4000 nM T20251 D05KUM 135446209 IC50 = 12589.25 nM T20251 D05LKO 44414722 IC50 = 22900 nM T20251 D05UZY 11539096 IC50 = 1600 nM T20251 D05VAB 9886249 IC50 = 100 nM T20251 D05VQJ 25147749 IC50 = 13240 nM T20251 D05XPV 54759259 IC50 > 25000 nM T20251 D05ZUX 44207909 IC50 = 20000 nM T20251 D06BMZ 46885513 IC50 > 65000 nM T20251 D06EMC 11392888 IC50 = 20000 nM T20251 D06HOI 44249821 IC50 > 80000 nM T20251 D06LJL 9916282 IC50 > 10000 nM T20251 D06MBD 11176403 IC50 = 8500 nM T20251 D06NXC 24996886 IC50 = 1460 nM T20251 D06NXK 46890563 Ki = 10000 nM T20251 D06QIQ 44592241 Ki = 3500 nM T20251 D07ADX 54764565 IC50 = 21000 nM T20251 D07ETF 9838960 Ki = 9599.99 nM T20251 D07GBV 10091189 Ki = 80 nM T20251 D07LFR 44231007 IC50 = 11000 nM T20251 D07SGS 44292136 IC50 = 130 nM T20251 D08CZT 9882067 Ki = 5700 nM T20251 D08EKQ 46890532 IC50 = 4950 nM T20251 D08JCU 44439386 Ki = 3900 nM T20251 D08NQA 57523213 IC50 = 12200 nM T20251 D08QBS 44178080 IC50 = 9500 nM T20251 D08RQW 49871766 Ki > 8000 nM T20251 D08TBU 15723 IC50 > 100000 nM T20251 D08ZIS 13007805 IC50 = 1600 nM T20251 D09BWE 11473281 IC50 > 30000 nM T20251 D09FGL 9910393 IC50 > 30000 nM T20251 D09FIC 46890395 IC50 = 10700 nM T20251 D09GZH 667538 IC50 = 810 nM T20251 D09HFT 44439376 Ki > 9000 nM T20251 D09KEB 11493841 IC50 = 3162.28 nM T20251 D09PTP 57325421 IC50 > 10000 nM T20251 D0A0GU 44247568 IC50 > 10000 nM T20251 D0A2BE 2780 IC50 = 602.56 nM T20251 D0A5KP 11588169 IC50 = 36000 nM T20251 D0A7GW 45487772 Ki = 12700 nM T20251 D0AT5N 56835134 IC50 = 16000 nM T20251 D0BD6A 10278617 IC50 > 30000 nM T20251 D0BW0V 44589528 IC50 = 1000 nM T20251 D0C2GE 67161540 IC50 = 3367 nM T20251 D0C2NK 4541 IC50 = 2290.87 nM T20251 D0C6BP 11567667 Ki = 8000 nM T20251 D0CM6T 11314340 IC50 = 13400 nM T20251 D0D6GI 46888441 IC50 > 10000 nM T20251 D0D8JU 46885546 IC50 > 60000 nM T20251 D0DA1E 23642319 Ki > 10000 nM T20251 D0DM6F 11761968 IC50 = 7000 nM T20251 D0E3DM 44592118 Ki = 15700 nM T20251 D0E7VO 59627005 IC50 > 32000 nM T20251 D0EG5G 46888467 IC50 > 10000 nM T20251 D0F9AM 86277846 Ki = 4.2 nM T20251 D0FF6S 16038374 IC50 > 30000 nM T20251 D0FJ1I 46891225 IC50 = 380 nM T20251 D0FL1D 9842124 Ki = 290 nM T20251 D0G4SU 65825 IC50 = 2500 nM T20251 D0G7LE 10991121 Ki = 1800 nM T20251 D0G8UA 46890321 IC50 > 10000 nM T20251 D0GG2J 46890492 IC50 = 760 nM T20251 D0H3GI 25129090 IC50 = 462 nM T20251 D0H8XV 12963076 IC50 = 900 nM T20251 D0I2UC 44230733 IC50 = 7000 nM T20251 D0J2YB 23631116 IC50 = 1600 nM T20251 D0JD4C 9853498 IC50 = 49900 nM T20251 D0K7RO 11646379 IC50 = 27500 nM T20251 D0L1UK 3064778 Ki = 7943.28 nM T20251 D0L9YP 44254503 IC50 = 11589 nM T20251 D0LM5H 11466357 EC50 = 8000 nM T20251 D0M1BJ 5282279 IC50 = 1500 nM T20251 D0N2DN 25129089 IC50 = 680 nM T20251 D0N2KU 44517677 IC50 > 20000 nM T20251 D0N6OL 11452268 IC50 = 10000 nM T20251 D0ND5D 10493741 Ki = 7000 nM T20251 D0O8AR 16097523 IC50 = 5200 nM T20251 D0OQ5H 46891330 IC50 = 40 nM T20251 D0OR6O 91623362 IC50 > 100000 nM T20251 D0P0QI 9816778 IC50 > 33000 nM T20251 D0P2HR 3510 IC50 = 3730 nM T20251 D0P6JS 11675054 IC50 = 16000 nM T20251 D0P7VQ 9929425 IC50 = 1000 nM T20251 D0P8PH 656732 IC50 > 32000 nM T20251 D0PC5A 44243144 IC50 = 30800 nM T20251 D0PC5N 71455 Ki > 150000 nM T20251 D0PF9Q 11472798 IC50 > 30000 nM T20251 D0Q8LS 11427736 IC50 = 2000 nM T20251 D0QG6A 9980734 IC50 = 43651.58 nM T20251 D0R0TW 11964036 IC50 > 20000 nM T20251 D0R3XC 11524350 Ki > 10000 nM T20251 D0R5OF 46885515 IC50 > 30000 nM T20251 D0RC9T 9795587 IC50 = 4897.79 nM T20251 D0S1XC 25224941 IC50 = 4400 nM T20251 D0S9AY 44592244 Ki = 8500 nM T20251 D0S9CI 11989776 Ki > 9000 nM T20251 D0SN6R 44592197 Ki > 5500 nM T20251 D0T4QX 11646823 IC50 = 1000 nM T20251 D0T9VC 56840673 IC50 > 10000 nM T20251 D0TO6S 2396 IC50 = 1000 nM T20251 D0U7OD 16043230 IC50 = 6950 nM T20251 D0UG5M 9956146 Ki = 8820 nM T20251 D0V0YM 24871527 IC50 = 1000 nM T20251 D0V3ZG 25192022 IC50 > 3000 nM T20251 D0V8DH 53380803 IC50 = 580 nM T20251 D0V8KA 42645487 IC50 = 33000 nM T20251 D0W2FU 53347902 IC50 > 30000 nM T20251 D0W3XD 16049828 Ki > 8000 nM T20251 D0W7WV 11039077 Ki = 61400 nM T20251 D0W8CA 46846313 IC50 < 2800 nM T20251 D0X7HD 11184481 IC50 = 40000 nM T20251 D0X8GC 45487773 Ki > 10000 nM T20251 D0XF5P 44592119 Ki = 16400 nM T20251 D0Y3OO 11327430 IC50 = 14000 nM T20251 D0Y4BL 11676971 IC50 > 10000 nM T20251 D0Y8AB 46885586 IC50 > 60000 nM T20251 D0Z7TM 22273644 IC50 = 6600 nM T20251 D0Z8PT 54758482 IC50 = 5000 nM T20251 D0ZC3Q 44230732 IC50 = 9000 nM T76059 D06OMK 445643 Ki = 0.4 nM T76059 D0G7UX 5284373 Ki = 20 nM T76059 D02VJY 3037617 IC50 = 17 nM T76059 D04PGB 445501 Ki = 0.01 nM T76059 D06GSE 9906804 Ki = 1 nM T76059 CA9GD5 3504 Ki = 7.5 nM T76059 CO43LW 444590 IC50 = 1.8 nM T76059 C5PE3Q 445644 Ki = 10 nM T76059 CU90XH 654676 Ki > 30000 nM T76059 COQ2J6 3154008 Ki > 50000 nM T76059 CR81OM 3154010 Ki = 33000 nM T76059 CW0TS4 3219611 Ki > 50000 nM T76059 CB9XT6 3219624 Ki > 50000 nM T76059 C14GPZ 3221232 Ki > 50000 nM T76059 C57KPB 3817957 Ki = 33000 nM T76059 CKE6R9 3827638 IC50 = 2600 nM T76059 CK18XS 4320284 Ki = 2500 nM T76059 CEX07C 4919428 Ki = 30000 nM T76059 CZ71ST 4921127 Ki = 37000 nM T76059 C2HUW7 5282071 EC50 = 1.6 nM T76059 CBMA23 5289261 Ki = 3.5 nM T76059 CTVP96 9798935 Ki = 2 nM T76059 C9M6IN 9798937 Ki = 820 nM T76059 CB92GZ 9801420 Ki = 8.9 nM T76059 CO7BG6 9806733 Ki = 54 nM T76059 C1PNB2 9809312 Ki = 19 nM T76059 CZ7GL8 9809998 IC50 = 9.6 nM T76059 CRD1T0 9811664 IC50 > 100000 nM T76059 C6NUY1 9817974 Ki = 8000 nM T76059 CTW24K 9819275 Ki = 20000 nM T76059 CYC61Z 9819945 Ki = 6000 nM T76059 C9IS6O 9820942 Ki = 130 nM T76059 C1XZ6E 9824296 Ki = 52 nM T76059 CX8W7L 9827812 IC50 = 16000 nM T76059 CW65IP 9841778 Ki = 1482 nM T76059 CK1VQ4 9845338 Ki = 6 nM T76059 CAU04E 9847345 Ki = 86 nM T76059 C8FAH3 9847925 Ki = 870 nM T76059 C12GZJ 9865798 Ki = 470 nM T76059 CS7LG9 9866557 Ki = 34 nM T76059 C2C1OB 9870251 IC50 = 200 nM T76059 C0EXC1 9870370 Ki = 105 nM T76059 C7JUR0 9871036 Ki = 3 nM T76059 C2NUK6 9873530 Ki = 0.3 nM T76059 C5VPL6 9883775 Ki = 35000 nM T76059 C6O4DI 9885558 IC50 = 4400 nM T76059 CS6F8D 9885875 Ki = 250 nM T76059 CZN2C1 9885966 Ki = 131 nM T76059 CAJ08L 9891805 Ki = 5 nM T76059 CV1PE8 9895267 Ki = 20 nM T76059 CFO6C1 9903902 Ki = 1300 nM T76059 CCJ0D9 9906857 Ki = 42 nM T76059 CSR87K 9908335 Ki = 72 nM T76059 C58ZLO 9909789 Ki = 504 nM T76059 CX09OR 9928246 Ki = 742 nM T76059 CNF68M 9934108 Ki = 25 nM T76059 C3V6MH 9936215 Ki = 50 nM T76059 CV4D7Y 9936936 Ki = 332 nM T76059 C37WXC 9938653 Ki = 1 nM T76059 CN4Z9I 9955490 Ki = 7 nM T76059 CZ37BG 9960384 Ki = 1 nM T76059 CH89YV 9962928 Ki = 1 nM T76059 CB26MR 9962976 Ki = 1 nM T76059 C3R1PD 9981138 Ki = 280 nM T76059 CX4T5W 10056711 Ki = 1.5 nM T76059 C3YFU6 10079556 Ki = 6 nM T76059 C67NVY 10102537 Ki = 9 nM T76059 CRYA61 10112806 Ki = 360 nM T76059 CTLA57 10114768 Ki = 123 nM T76059 C0H6TX 10118511 Ki = 591 nM T76059 C7Y9UG 10138683 Ki = 420 nM T76059 C08VEM 10140711 Ki = 590 nM T76059 C03BSX 10155516 Ki = 12.2 nM T76059 C4CE6L 10161454 Ki = 104 nM T76059 C52TDP 10161566 Ki = 210 nM T76059 CIQH49 10161855 Ki = 150 nM T76059 C5PGQ8 10177566 Ki = 8.7 nM T76059 CV4IK3 10183195 Ki = 360 nM T76059 C0Y4IK 10183484 Ki = 82 nM T76059 CQN3P4 10198461 Ki > 10000 nM T76059 C8R5DX 10229698 Ki = 88 nM T76059 C7B0JO 10229811 Ki = 92 nM T76059 CS9HP2 10234693 Ki = 1 nM T76059 C57GIZ 10259637 IC50 = 0.77 nM T76059 C8DLF4 10260436 Ki = 38 nM T76059 C4RW1L 10260525 Ki = 7 nM T76059 C7GJ6Y 10276095 Ki = 84 nM T76059 C6GVC7 10301493 Ki = 640 nM T76059 CU7D3Z 10303855 Ki = 156 nM T76059 C2YUE4 10317191 Ki = 550 nM T76059 CSN72K 10371065 IC50 = 114 nM T76059 C4XD1F 10396050 Ki = 1 nM T76059 C1HOM8 10396073 IC50 = 2.9 nM T76059 CI4FP1 10396108 Ki = 10 nM T76059 C4O6QS 10463260 IC50 = 0.6 nM T76059 CZ0S3I 10463451 Ki = 29 nM T76059 CJ0LZ4 10474617 Ki = 11 nM T76059 CDFQ06 10486039 Ki = 3 nM T76059 CF3GI4 10508532 Ki = 900 nM T76059 CSIR58 10555604 IC50 = 40 nM T76059 CLOT05 10571272 IC50 = 116700 nM T76059 C6WJG4 10574954 Ki = 350 nM T76059 C0P3TN 10587060 Ki = 83000 nM T76059 C7F9PD 10618401 Ki = 570 nM T76059 CWDG54 10619661 Ki = 14000 nM T76059 C3IAZ8 10623440 Ki = 390 nM T76059 CR4IY5 10626978 IC50 = 1530 nM T76059 CC5DF2 10640341 Ki = 790 nM T76059 CL4C8T 10664741 IC50 = 21600 nM T76059 CE8TZ1 10668143 Ki = 370 nM T76059 CH9AV3 10685294 IC50 = 124100 nM T76059 C35GOE 10687366 IC50 > 200000 nM T76059 C1G6BY 10689335 Ki = 6500 nM T76059 CSO83D 10714474 Ki = 150 nM T76059 C12HRN 10715720 IC50 = 22300 nM T76059 CEVL01 10732772 IC50 = 3100 nM T76059 CF2A9U 10734201 Ki = 7200 nM T76059 C8TG7O 10741010 Ki = 220 nM T76059 CSYB76 10756782 Ki = 67000 nM T76059 C1K6HQ 10758826 Ki = 24000 nM T76059 CZ2OR8 10790307 Ki = 200 nM T76059 C63LIX 10834562 IC50 = 68200 nM T76059 C9TQ7U 11105029 EC50 = 21.1 nM T76059 C5NB9Z 11129344 IC50 = 17100 nM T76059 CO2RJ8 11181229 Ki = 137000 nM T76059 CZ29YS 11742535 Ki = 120 nM T76059 C0RHG3 11792025 Ki = 8400 nM T76059 CA1JR7 11800691 IC50 > 200000 nM T76059 CGR93V 11851094 Ki = 34 nM T76059 CR2BC8 11851095 Ki = 34 nM T76059 C58HTG 15380464 Ki = 725 nM T76059 C9VHU1 15380465 Ki = 130 nM T76059 C5WJK3 15380466 Ki = 30 nM T76059 CBG7J0 15380467 Ki = 60 nM T76059 C6UX1B 15380469 Ki = 12 nM T76059 C1O3HC 15380471 Ki = 20 nM T76059 CJ27ZQ 15380472 Ki = 103 nM T76059 CZI61J 15380473 Ki = 760 nM T76059 CGDE51 15380474 Ki = 210 nM T76059 CY4E8J 15380475 Ki = 32 nM T76059 C8IK5U 15380476 Ki = 24 nM T76059 CO0MS8 15516000 Ki = 110 nM T76059 C0S5YD 15545973 IC50 = 15 nM T76059 C7WJF0 15546641 EC50 = 9.2 nM T76059 C94PQN 16394002 Ki = 1500 nM T76059 CDK6Q3 16485668 Ki = 7600 nM T76059 CG12OR 20707827 Ki = 3 nM T76059 C6K9WT 20725894 Ki = 0.5 nM T76059 CW2F6L 21027754 Ki = 450 nM T76059 C0S5GA 21027755 Ki = 250 nM T76059 C9Y0RT 21027758 Ki = 18 nM T76059 CGA08F 21027759 Ki = 82 nM T76059 CH8C9X 21258251 Ki = 170 nM T76059 CFJ0N7 21258256 Ki = 13 nM T76059 COI19B 21363697 Ki = 143 nM T76059 C3C9LX 21363707 Ki = 54 nM T76059 CYT86D 21363714 Ki = 217 nM T76059 CEA2K3 22064769 Ki > 10000 nM T76059 CY4R0O 23555949 Ki = 42 nM T76059 CHG49U 24860365 Ki = 69 nM T76059 CH8EQ3 24860366 Ki = 85 nM T76059 C3C1RK 24860367 Ki = 126 nM T76059 CVU23R 24860368 Ki = 152 nM T76059 CWB04A 24860369 Ki = 171 nM T76059 C2JL4P 24860370 Ki = 201 nM T76059 CR0OU1 24860371 Ki = 225 nM T76059 CQ6K8G 24860372 Ki = 46 nM T76059 CTB24N 24860373 Ki = 60 nM T76059 CCXP98 24860374 Ki = 71 nM T76059 CKY5C1 24860375 Ki = 72 nM T76059 C83GJK 24860376 Ki = 100 nM T76059 C6SD1K 24860377 Ki = 110 nM T76059 C2LK7D 24860378 Ki = 123 nM T76059 C87AXJ 24860379 Ki = 131 nM T76059 CM3F2Y 24860380 Ki = 238 nM T76059 C0D4FK 24860381 Ki = 282 nM T76059 CQZ9I6 24860382 Ki = 583 nM T76059 CRZ43B 24860383 Ki = 586 nM T76059 CZ85UH 24860384 Ki = 1000 nM T76059 CK29UW 24860385 Ki = 153 nM T76059 C7I6EL 24860386 Ki = 20800 nM T76059 C61YFI 24860387 Ki = 208 nM T76059 CQIG36 24860388 Ki = 3100 nM T76059 C1V8WX 24860389 Ki = 91 nM T76059 CH3P2O 24860390 Ki = 31700 nM T76059 C5U9FE 24860391 Ki = 107 nM T76059 C63IOV 24860392 Ki = 110 nM T76059 C6IXT3 24860393 Ki = 114 nM T76059 CBKW67 24860394 Ki = 279 nM T76059 CJ73FA 24860395 Ki = 2300 nM T76059 C09HAI 24860396 Ki = 244 nM T76059 C6PFH1 24860397 Ki = 266 nM T76059 C5JY0D 24860398 Ki = 288 nM T76059 C84WFH 24860402 Ki = 183 nM T76059 CNLZ96 24860403 Ki = 236 nM T76059 CTLC58 35027274 IC50 = 100 nM T76059 CBX15K 42897553 Ki = 4700 nM T76059 CV1SX2 44265409 EC50 = 12 nM T76059 CBX13N 44269758 IC50 = 1.5 nM T76059 C6OUP3 44269765 IC50 = 19 nM T76059 CR9J7V 44269773 IC50 = 65 nM T76059 C2YM7N 44269774 IC50 = 126 nM T76059 C1Y8AV 44269775 IC50 = 94 nM T76059 CI27YN 44269786 IC50 = 273 nM T76059 CG5H3K 44269787 IC50 = 5.8 nM T76059 CM9EC2 44269801 IC50 = 133 nM T76059 CXYL79 44269804 IC50 = 590 nM T76059 C3RF5Y 44269806 IC50 = 4.4 nM T76059 CO5N4A 44269817 IC50 = 12 nM T76059 CUKA34 44269842 IC50 = 150 nM T76059 CDX04K 44269845 IC50 = 187 nM T76059 C0KXL4 44269846 IC50 = 43 nM T76059 C96LNO 44269847 IC50 = 3.8 nM T76059 CKEL40 44269849 IC50 = 19 nM T76059 CU5LH8 44269870 IC50 = 66 nM T76059 C6SN3J 44279552 IC50 > 1000 nM T76059 C18XMQ 44279663 IC50 > 1000 nM T76059 CBS95E 44279849 IC50 = 14 nM T76059 C1RAK8 44280039 Ki = 3.7 nM T76059 C69FGM 44280289 IC50 = 2.1 nM T76059 CYNR42 44280488 Ki > 10000 nM T76059 CYV0B7 44280537 Ki = 3100 nM T76059 CA29IB 44280566 Ki = 5200 nM T76059 C0ZX7Y 44280567 Ki = 6000 nM T76059 CFT18Q 44280568 Ki = 4400 nM T76059 CI47SZ 44280581 Ki = 7200 nM T76059 CUVJ79 44280582 Ki = 47000 nM T76059 C24LTB 44280606 Ki = 18000 nM T76059 C0WL4I 44280742 Ki = 420 nM T76059 C7WQH2 44280751 Ki = 480 nM T76059 CL8FN0 44280766 Ki = 320 nM T76059 CWHU46 44280776 Ki = 8000 nM T76059 C67YOK 44280790 Ki = 4400 nM T76059 CSKB97 44280791 Ki = 1400 nM T76059 CP6N8F 44280797 Ki = 3800 nM T76059 C0K8IC 44280799 Ki = 1300 nM T76059 C8VZY0 44280800 Ki = 12 nM T76059 CILS94 44280811 Ki = 86 nM T76059 C5G8JO 44280833 Ki = 32 nM T76059 C6C2KX 44280834 Ki = 2100 nM T76059 C6A0WV 44280845 Ki = 260 nM T76059 C8I9HQ 44280846 Ki = 2700 nM T76059 C7GN1W 44280850 Ki = 1500 nM T76059 CN2PS9 44280851 Ki = 850 nM T76059 C48DQA 44280852 Ki = 22 nM T76059 CN45YP 44280871 Ki = 1300 nM T76059 C0H6RY 44280888 Ki = 1000 nM T76059 C9N1YQ 44280917 Ki = 2300 nM T76059 CB1OE4 44280918 Ki = 47 nM T76059 C6UO7I 44280919 Ki = 740 nM T76059 CN9I3W 44280941 Ki = 1200 nM T76059 CK27HI 44280958 Ki > 50000 nM T76059 CFW93J 44280959 Ki > 50000 nM T76059 C56KBA 44281035 Ki = 400 nM T76059 CV1B3D 44281045 Ki = 120 nM T76059 C54BJK 44281046 Ki = 220 nM T76059 CS26ZL 44281058 Ki = 470 nM T76059 C7BIA5 44281072 Ki = 92 nM T76059 C43DEQ 44281082 Ki = 180 nM T76059 CCG2H5 44281092 Ki = 1200 nM T76059 CM96EN 44281103 Ki = 720 nM T76059 CXTP68 44281114 Ki > 50000 nM T76059 CO0VR5 44281130 Ki = 1300 nM T76059 CADL82 44281131 Ki = 22000 nM T76059 CKUR12 44281153 Ki > 50000 nM T76059 CLOF28 44281158 Ki = 820 nM T76059 C3OF7W 44281160 Ki = 9500 nM T76059 C6M8JF 44281206 Ki > 50000 nM T76059 CHG02K 44281207 Ki > 50000 nM T76059 C8UI7Y 44281208 Ki = 1100 nM T76059 CT69UY 44281209 Ki = 2400 nM T76059 CANW36 44281215 Ki = 32000 nM T76059 CJET58 44281216 Ki = 42000 nM T76059 COY8M2 44281230 Ki = 22000 nM T76059 CCJ91K 44281233 Ki = 2800 nM T76059 C5OJQ2 44281249 Ki > 50000 nM T76059 CJL61F 44281259 Ki > 50000 nM T76059 CWO5Q9 44281260 Ki > 50000 nM T76059 CDB38P 44281261 Ki = 24000 nM T76059 C1D9BI 44281262 Ki = 6300 nM T76059 CD2QG9 44281272 Ki = 5400 nM T76059 CV7TY3 44281280 Ki > 33000 nM T76059 C61NZB 44281286 Ki = 3900 nM T76059 CD7UC9 44281293 Ki > 50000 nM T76059 CO5E0F 44281298 Ki = 1300 nM T76059 COX6I8 44281299 Ki = 11000 nM T76059 CM7OB4 44281311 Ki = 13000 nM T76059 C65VBK 44281361 Ki = 640 nM T76059 C7WFB3 44281383 Ki = 1600 nM T76059 CPL10S 44281410 Ki = 1600 nM T76059 CP2RU7 44281411 Ki = 110 nM T76059 CHA8T5 44281412 Ki = 2200 nM T76059 C0WNT3 44281413 Ki = 13000 nM T76059 CZQC70 44281458 Ki > 50000 nM T76059 CP2K6S 44281459 Ki = 1400 nM T76059 CY36QT 44281487 Ki = 4200 nM T76059 CO57JP 44281695 Ki = 39000 nM T76059 CRG59M 44281696 Ki > 50000 nM T76059 C4RGM1 44287122 Ki = 207 nM T76059 CS3O2T 44294553 IC50 = 3.3 nM T76059 CFHW79 44294716 IC50 = 13 nM T76059 C8CM5N 44294717 IC50 = 5.6 nM T76059 C48QMD 44294726 IC50 = 2.4 nM T76059 CK3OQ4 44294727 IC50 = 2 nM T76059 CQ4G9T 44294866 IC50 = 470 nM T76059 C7V1GU 44294867 IC50 = 50 nM T76059 C0K7FS 44294868 IC50 = 180 nM T76059 C8DZ7M 44294869 IC50 = 500 nM T76059 CT36GW 44294871 IC50 = 9.4 nM T76059 CV65SR 44294876 IC50 = 46 nM T76059 CO0TL9 44294886 IC50 = 16 nM T76059 CSW9I5 44294887 IC50 = 3.2 nM T76059 CT7PM2 44294894 IC50 = 4 nM T76059 CN6AB9 44294895 IC50 = 170 nM T76059 CR0YF6 44294896 IC50 = 19 nM T76059 C8KJL3 44294897 IC50 = 71 nM T76059 CBZ7G2 44294938 IC50 = 180 nM T76059 CSBI84 44294939 IC50 = 570 nM T76059 CYL6X0 44294966 IC50 = 48 nM T76059 C3WK8M 44294990 IC50 = 0.4 nM T76059 CF8R6K 44295208 IC50 = 68 nM T76059 C1C9TW 44295523 Ki = 8.3 nM T76059 CU2A6K 44306123 EC50 = 18 nM T76059 C7WNM2 44306124 EC50 = 12 nM T76059 C86EOZ 44306135 EC50 = 13.6 nM T76059 C8T5NI 44306145 EC50 = 32 nM T76059 CF75NO 44306146 EC50 = 5.3 nM T76059 CUH17I 44306155 EC50 = 9 nM T76059 C6OQ4D 44306156 EC50 = 45 nM T76059 CN58YR 44306157 EC50 = 7.5 nM T76059 C8N7QZ 44306253 EC50 = 45 nM T76059 CD8O6N 44306280 EC50 = 7.5 nM T76059 C68IRQ 44306324 EC50 = 11.25 nM T76059 C46AQD 44309746 IC50 = 1.6 nM T76059 C72NFI 44309747 IC50 = 3.6 nM T76059 CTI60L 44309800 IC50 = 10 nM T76059 CMC52Q 44309855 IC50 = 74.8 nM T76059 COH7M3 44309856 IC50 = 5.1 nM T76059 C24URG 44309955 IC50 = 0.8 nM T76059 C1CD5Q 44309983 IC50 = 2.8 nM T76059 CZN4T6 44309984 IC50 = 0.7 nM T76059 C2C9GA 44312111 EC50 = 30 nM T76059 CW5ZR8 44312113 EC50 = 22 nM T76059 CO56DC 44312417 EC50 = 20.5 nM T76059 CER3Y9 44312559 EC50 = 7.4 nM T76059 CQ5H2I 44312595 EC50 = 12 nM T76059 CKO38Y 44337706 IC50 = 64 nM T76059 C4QJC3 44337851 IC50 = 26 nM T76059 CM38LX 44337859 IC50 = 12 nM T76059 CF4VZ3 44337877 IC50 = 8.2 nM T76059 C6V5LW 44337938 IC50 = 5.5 nM T76059 CP0U7C 44338501 IC50 = 200 nM T76059 C64ZIF 44340105 Ki = 175 nM T76059 C3FV8H 44340118 Ki = 190 nM T76059 CIS1X4 44340142 Ki = 5 nM T76059 CFR52J 44340151 Ki = 340 nM T76059 CU3O2I 44340152 Ki = 190 nM T76059 CLFQ54 44340165 Ki = 25 nM T76059 CK1A4T 44340166 Ki = 5 nM T76059 C5KSH2 44340326 Ki > 5000 nM T76059 C4D5TV 44340429 Ki = 6000 nM T76059 CKP76I 44340465 Ki = 400 nM T76059 C4KI2O 44340482 Ki = 130 nM T76059 CHV95O 44350652 Ki = 8100 nM T76059 CKQU96 44350663 Ki = 8300 nM T76059 C24PEN 44350671 Ki = 1500 nM T76059 CND94Q 44350709 Ki > 50000 nM T76059 C0YXR3 44350766 Ki = 1200 nM T76059 CZ6D5G 44350783 Ki = 10000 nM T76059 CJ6HO2 44360860 IC50 = 3.4 nM T76059 C0F3WL 44365027 Ki = 195 nM T76059 CXGI06 44365035 Ki = 12 nM T76059 CCA08O 44365058 Ki = 170 nM T76059 CVT27W 44365059 Ki = 120 nM T76059 CF97ST 44365150 Ki = 3 nM T76059 CNFK71 44365151 Ki = 95 nM T76059 CG96PA 44365152 Ki = 9 nM T76059 C2MQ1T 44365238 Ki = 70 nM T76059 C4RD0I 44365240 Ki = 116 nM T76059 CZ1QB9 44365271 Ki = 17 nM T76059 C50CGS 44365344 Ki = 78 nM T76059 C47LAT 44365384 Ki > 10000 nM T76059 C6FI7B 44365447 Ki = 107 nM T76059 CK0YA4 44365450 Ki = 194 nM T76059 CI59UY 44365487 Ki = 40 nM T76059 CSH76C 44365490 Ki = 17 nM T76059 CLBE84 44365587 Ki = 15 nM T76059 C5FR3M 44368603 Ki = 32 nM T76059 CRTX63 44368604 IC50 = 410 nM T76059 C0HB4I 44368605 Ki = 482 nM T76059 CJZ6I1 44368744 Ki = 1300 nM T76059 CAR35L 44383333 EC50 = 34.3 nM T76059 CZ50YE 44383482 EC50 = 23 nM T76059 C1FED5 44383746 EC50 = 12 nM T76059 CB1P6R 44383908 EC50 = 11.8 nM T76059 C8R5WF 44383962 EC50 = 6.1 nM T76059 C6T4NQ 44384095 EC50 = 5.7 nM T76059 C79TFY 44384115 EC50 = 2.7 nM T76059 CE0X3V 44384116 EC50 = 6.6 nM T76059 CVM90W 44384124 EC50 = 9.2 nM T76059 CV19BZ 44384125 EC50 = 7 nM T76059 CSG64P 44384126 EC50 = 14.9 nM T76059 C65GRN 44384267 EC50 = 3.4 nM T76059 C02QJT 44385122 EC50 = 10.3 nM T76059 CQH7N8 44385184 EC50 = 15.6 nM T76059 C0TJ7O 44385185 EC50 = 4.6 nM T76059 CXA4S0 44387197 Ki = 250 nM T76059 CP96AN 44407027 Ki = 330 nM T76059 CKR3O4 44407127 Ki = 7000 nM T76059 C78BIN 44407142 Ki = 2700 nM T76059 CMUE21 44407218 Ki = 357 nM T76059 CZD8Y4 44407219 Ki = 772 nM T76059 CMY5V3 44461925 Ki = 210 nM T76059 C7YWU8 44461941 Ki = 2.8 nM T76059 CQA89Y 44461954 Ki = 112 nM T76059 C9JN0R 44461955 Ki = 258 nM T76059 CG51ZB 44461956 Ki = 68 nM T76059 CN68YV 44461964 Ki = 81 nM T76059 C7SZ3Q 50994120 IC50 > 30000 nM T76059 CX6PV4 50994121 IC50 = 2800 nM T76059 CY5FL8 50994123 IC50 > 30000 nM T76059 CNZ46O 50994197 IC50 = 4200 nM T76059 CGQF17 50994198 IC50 = 120 nM T76059 CBIR56 50994199 IC50 = 150 nM T76059 C4T1YW 50994200 IC50 = 70 nM T76059 CU51AK 50994201 IC50 = 320 nM T76059 CD3X0R 50994202 IC50 = 260 nM T76059 CID87X 51049455 Ki = 4.5 nM T76059 C2V6RJ 56962328 IC50 = 130 nM T76059 CJ46RD 56962330 IC50 = 343 nM T76059 C1BUW4 57521458 IC50 = 510 nM T76059 CGU89M 57521460 IC50 = 2450 nM T76059 CKP31Q 57521461 IC50 = 100 nM T76059 C7D3PN 57521557 IC50 = 1050 nM T76059 CO6T0F 57521558 IC50 = 150 nM T76059 C2RVN0 57521777 IC50 = 60 nM T76059 C8PY2R 57521778 IC50 = 50 nM T76059 C0HOD9 57521879 IC50 = 50 nM T76059 CS7B2A 57521880 IC50 = 60 nM T76059 CGP03D 57521881 IC50 = 1800 nM T76059 C9V4QB 57521882 IC50 = 1200 nM T76059 C4C7LK 57522005 IC50 = 1100 nM T76059 C8YI0U 57522006 IC50 = 10100 nM T76059 C0KC6J 57522007 IC50 = 4600 nM T76059 CH89PN 57522008 IC50 = 3800 nM T76059 CG6TK3 57522120 IC50 = 1900 nM T76059 CWQ8J7 57522121 IC50 = 1900 nM T76059 CTCH51 57522237 IC50 = 1090 nM T76059 C8R2IJ 57522238 IC50 = 320 nM T76059 C1PBX3 57522239 IC50 = 800 nM T76059 CU5NP7 57522240 IC50 = 6100 nM T76059 C0P3TI 57522347 IC50 = 7600 nM T76059 C6WY9D 57522348 IC50 = 600 nM T76059 CM7ZV1 57522349 IC50 = 1000 nM T76059 C6FQ4X 57522350 IC50 = 5100 nM T76059 CHVK79 57522455 IC50 = 2400 nM T76059 C73XQS 57522456 IC50 = 4500 nM T76059 C4OJX2 57522457 IC50 = 670 nM T76059 CGIX69 57522458 IC50 = 230 nM T76059 CG2SO6 57522567 IC50 = 1180 nM T76059 CR9C3F 57522569 IC50 = 1500 nM T76059 C8SP3L 57522570 IC50 = 2570 nM T76059 CQ3I7G 57522682 IC50 = 1200 nM T76059 C5QM2O 57522683 IC50 = 21 nM T76059 CE7G2U 57522684 IC50 = 660 nM T76059 CA4R9I 57522685 IC50 = 750 nM T76059 C3EP9M 57522800 IC50 > 100000 nM T76059 C46EIF 57522801 IC50 = 200 nM T76059 CC85GJ 57522802 IC50 > 50000 nM T76059 CCUW31 57522803 IC50 > 50000 nM T76059 CV58SP 57522927 IC50 = 800 nM T76059 CT58KB 57522928 IC50 = 115 nM T76059 C95OGY 57522929 IC50 > 50000 nM T76059 CZI07G 57522930 IC50 = 3 nM T76059 C8B9HE 57522931 IC50 = 450 nM T76059 C7Y9SK 57523063 IC50 = 550 nM T76059 C4S5KW 57523064 IC50 = 1290 nM T76059 CT4NB0 57523068 IC50 > 100000 nM T76059 C0NUH8 57523069 IC50 = 1400 nM T76059 C2YN0S 57523070 IC50 = 870 nM T76059 CG5AB2 57783590 IC50 = 6.8 nM T76059 C2DIM5 70684253 IC50 = 3380 nM T76059 CYQH64 70684260 IC50 = 470 nM T76059 CG5D2W 70688508 IC50 = 2200 nM T76059 CWDU09 70688522 IC50 = 570 nM T76059 C14GSV 70690624 EC50 = 5 nM T76059 CWY7C0 70692710 IC50 = 310 nM T76059 CF34ES 70694690 Ki = 0.7 nM T76059 C5MK3W 70694725 IC50 = 8100 nM T76059 CD65LN 70694726 IC50 = 9100 nM T76059 CEZG14 70694756 IC50 = 2780 nM T76059 CU9RN3 70694757 IC50 = 60 nM T76059 CRWB36 71718375 Ki = 2800 nM T76059 C61TIG 71718376 Ki = 870 nM T76059 CR9FQ3 71718981 Ki = 500 nM T76059 CK36QR 71720180 Ki = 2100 nM T76059 CUT2Y6 71720824 Ki = 27700 nM T76059 C0H2QE 73345516 Ki = 50 nM T76059 C5EMH2 86277875 Ki = 90 nM T76059 CXF34A 89939931 Ki = 8.8 nM T76059 C29TEF 101167236 Ki = 4000 nM T76059 CCH84L 117967740 Ki = 23400 nM T76059 CXP8S2 117967763 Ki = 2000 nM T76059 CEY28F 117967783 Ki = 12400 nM T76059 C46GRQ 117967787 Ki = 3800 nM T76059 C2A8EM 117967798 Ki = 12100 nM T76059 CVP4Q3 117967801 Ki = 120000 nM T76059 CWTL26 117967814 Ki = 1000 nM T76059 C5GF3N 117967822 Ki = 51900 nM T76059 CJ26YR 117967829 Ki = 30700 nM T76059 C2AF1T 117967843 Ki = 3200 nM T76059 CRCH91 117967851 Ki = 26900 nM T76059 CT3DQ5 117967872 Ki = 71100 nM T76059 C7NTU4 117967885 Ki = 50300 nM T76059 CYS70L 117967909 Ki = 101000 nM T76059 CU86WK 117967913 Ki = 6000 nM T76059 CFA74P 117967937 Ki = 10900 nM T76059 C08BKM 117967939 Ki = 11500 nM T76059 CHN52K 117967946 Ki = 5600 nM T76059 C1ZYL4 117967947 Ki = 1200 nM T76059 CA6ZJ7 117967955 Ki = 317000 nM T76059 C2QZ3D 117967964 Ki = 6600 nM T76059 C07HJM 117967978 Ki = 22500 nM T76059 CSD64M 117968002 Ki = 6600 nM T76059 CTI1X7 117968005 Ki = 6800 nM T76059 CXP8N7 117968006 Ki = 4300 nM T76059 C4LAX1 117968012 Ki = 8700 nM T76059 C58LQV 117968031 Ki = 30100 nM T76059 CF1GO9 117968050 Ki > 300000 nM T76059 CXLE07 117968053 Ki = 7500 nM T76059 CXWU20 117968117 Ki = 46900 nM T76059 CZQB61 117968118 Ki = 12800 nM T76059 CG65FE 117968136 Ki = 25100 nM T76059 C5O7SB 117968142 Ki = 39700 nM T76059 C5EU1T 117968149 Ki = 49200 nM T76059 CEXT51 117975049 Ki = 3000 nM T76059 CELN63 118233557 IC50 = 14.3 nM T76059 CJ84MI 118233582 IC50 = 9.52 nM T76059 CBP3S9 118233586 IC50 = 13.39 nM T76059 CUW1S0 118233596 IC50 = 12.61 nM T76059 CNP23H 122192627 Ki = 600 nM T76059 CEMN03 122192628 Ki = 1200 nM T76059 C5ZF3W 122192629 Ki = 300 nM T76059 CG2U4V 122693787 IC50 = 11.19 nM T76059 CPJ47S 122693793 IC50 = 12.48 nM T76059 C4YI9N 122693794 IC50 = 824 nM T76059 CC0L6K 127024999 Ki = 22300 nM T76059 C0SKD7 127053468 Ki = 4200 nM T76059 CHSY35 137631778 Ki = 7 nM T76059 CQ9F8R 137632505 IC50 = 10.99 nM T76059 C86IDH 137633267 Ki = 11.8 nM T76059 CWM7H1 137634012 Ki = 49 nM T76059 CGWE89 137639136 Ki = 249 nM T76059 C35SVI 137639141 Ki = 7 nM T76059 CAI70F 137640680 Ki = 21.1 nM T76059 CAM69O 137642452 Ki = 49 nM T76059 COK87T 137642715 IC50 = 19.2 nM T76059 C1P6LO 137642835 Ki = 0.45 nM T76059 CKL06A 137645398 IC50 = 23.6 nM T76059 C8DKV2 137649029 Ki = 7 nM T76059 C4IRT9 137649504 Ki = 49 nM T76059 C0EQ5V 137649552 Ki = 18.8 nM T76059 C9N2BM 137649843 IC50 = 27 nM T76059 CXSK64 137650264 Ki = 49 nM T76059 C93ENA 137650602 IC50 = 22.1 nM T76059 C7LYA9 137652507 Ki = 49 nM T76059 CC3LT2 137652724 IC50 = 19.1 nM T76059 CRLW34 137656432 IC50 = 12.59 nM T76059 CQR9J3 137657364 Ki = 143 nM T76059 CM05LU 137658940 Ki = 7 nM T76059 CHK6O9 137660768 Ki = 7 nM T76059 C8DI6S 137661451 IC50 = 22.6 nM T76059 CMA0I1 145980548 Ki = 5 nM T76059 C24MVU 145981935 Ki = 7 nM T76059 C6Z4QJ 145982171 IC50 = 53.6 nM T76059 CIRN21 145988906 Ki = 1 nM T76059 CP16HY 145989176 IC50 = 800 nM T76059 C61QME 155547348 Ki = 210 nM T76059 CGA13H 44287121 Ki = 400 nM T76059 D06ZWX 6197 Ki = 3400 nM T00663 D02NNV 3038525 IC50 > 5000 nM T00663 D02ZQS 16095342 IC50 > 10000 nM T00663 D03LWG 53235510 IC50 > 10000 nM T00663 D07EHV 44814409 IC50 > 10000 nM T00663 D0A6VD 25073775 IC50 = 160 nM T00663 D0HY9S 73386890 IC50 = 242 nM T00663 D0X4MN 11597537 IC50 = 6 nM T00663 D03BNU 59604787 IC50 > 10000 nM T00663 D05SJB 10040667 IC50 = 32 nM T00663 D08DNZ 45102739 IC50 = 11 nM T00663 D0PG5N 25123232 IC50 = 7750 nM T00663 D0UY9Y 46869000 IC50 = 800 nM T00663 D0W7MG 11647397 IC50 = 210 nM T00663 D0W8BL 46868926 IC50 = 9 nM T00663 D0ZU8L 57340689 IC50 = 9 nM T00663 D0F8DL 176155 Ki = 90 nM T00663 D0T3ME 156422 IC50 = 1400 nM T00663 C9W4UM 290221 IC50 = 1500 nM T00663 C5DB6Y 447872 IC50 = 1.6 nM T00663 C3V0TX 447873 IC50 = 1.6 nM T00663 C9VW8M 449054 IC50 > 16000 nM T00663 CKG76T 579429 IC50 = 3162.28 nM T00663 C0EQ6J 622378 IC50 > 15848.93 nM T00663 C2Y0RL 626628 IC50 > 15848.93 nM T00663 CQ9PB5 684674 IC50 > 15848.93 nM T00663 CR93CZ 746075 IC50 = 1830 nM T00663 CK89TF 766948 IC50 = 398.11 nM T00663 CWO49I 826287 IC50 > 15848.93 nM T00663 CVY4C5 847353 IC50 > 15848.93 nM T00663 CKS84B 897877 IC50 = 1000 nM T00663 CG2BU0 921636 Ki > 10000 nM T00663 C3PBJ1 942437 IC50 = 31800 nM T00663 C6K8WV 979869 IC50 = 1100 nM T00663 C4XP1N 1100747 IC50 = 3162.28 nM T00663 C8HP2S 1208196 IC50 = 2430 nM T00663 CG0IU6 1228584 IC50 = 1900 nM T00663 CRGB47 1228713 IC50 = 620 nM T00663 CV9D8Y 1228716 IC50 = 350 nM T00663 C67OWG 1228882 IC50 = 590 nM T00663 C5F4WM 1473242 Ki > 4000 nM T00663 C0VQG3 1483690 Ki = 13000 nM T00663 C2EX5Q 1641795 IC50 = 6570 nM T00663 CLBQ01 1737773 IC50 = 750 nM T00663 C5VE3K 2231029 IC50 = 1700 nM T00663 CF8Z5H 2766666 Ki = 5200 nM T00663 CQN85O 2766806 Ki = 9900 nM T00663 C8UC4F 2766824 Ki = 5000 nM T00663 C7IF4L 2766825 Ki = 6700 nM T00663 CZHL80 2808202 IC50 = 2200 nM T00663 CW6P5E 2823737 IC50 > 15848.93 nM T00663 C3KEG9 2823738 IC50 = 10000 nM T00663 C8WSF5 3659633 IC50 = 559 nM T00663 CR0DJ8 4078145 IC50 = 40 nM T00663 C69GSP 4079571 IC50 = 2700 nM T00663 CW26HV 5337145 IC50 = 14190 nM T00663 CSFQ07 9549178 IC50 = 3 nM T00663 CN8K3H 9814292 IC50 = 950 nM T00663 C7Q6PF 9818586 Ki = 720 nM T00663 C71GHF 9826147 IC50 > 10000 nM T00663 CW8V0K 9864418 IC50 > 16000 nM T00663 COR3S2 9892736 IC50 = 150 nM T00663 CX5G3A 9928616 IC50 = 30 nM T00663 CN0AJ9 9934347 IC50 = 12 nM T00663 C0V7UW 9958506 IC50 = 30 nM T00663 CO4B8A 9982333 IC50 > 10000 nM T00663 C37GXK 9983303 IC50 > 16000 nM T00663 C93OCY 10021870 IC50 = 175 nM T00663 C4PRY1 10066845 IC50 = 18 nM T00663 C2C1BP 10089048 IC50 > 16000 nM T00663 CLA50K 10091293 IC50 = 33 nM T00663 CPN3T4 10092520 IC50 = 32 nM T00663 CBJU36 10093433 IC50 = 26 nM T00663 CF1P3X 10094511 IC50 = 28500 nM T00663 C9NO1X 10149689 IC50 = 202 nM T00663 CYE4T2 10151272 IC50 = 21 nM T00663 CN0QK4 10152189 IC50 = 3.4 nM T00663 C69DHW 10158652 IC50 < 16000 nM T00663 CR47IV 10172440 IC50 = 32 nM T00663 CQU9K5 10200651 Ki > 4000 nM T00663 C7QHS0 10215642 IC50 = 5.3 nM T00663 C9PFR4 10225532 IC50 = 61.2 nM T00663 C1I0SL 10247954 IC50 = 7 nM T00663 C9NJ1X 10269964 IC50 = 70 nM T00663 C7SFI1 10296883 IC50 > 10000 nM T00663 CB59MP 10310219 IC50 = 1.9 nM T00663 CFL5O8 10364826 IC50 = 15 nM T00663 C72AVO 10372770 IC50 = 500 nM T00663 C2G3YH 10384284 IC50 = 652 nM T00663 CJE04Q 10384407 IC50 = 108 nM T00663 CFD01W 10452031 IC50 = 17 nM T00663 CB0E2X 10472936 IC50 = 20 nM T00663 CT92AO 10475988 IC50 = 528 nM T00663 CRBL32 10477561 IC50 = 693 nM T00663 CRX6F0 10479082 IC50 > 16000 nM T00663 CB47LY 10847715 IC50 > 15848.93 nM T00663 CIB8M9 11353316 IC50 = 10000 nM T00663 C0APW4 11422034 IC50 = 70 nM T00663 CMI8G3 11478147 IC50 = 13000 nM T00663 CJ9OH7 11538129 IC50 = 410 nM T00663 CTG83F 11539329 Ki = 72 nM T00663 CACS26 11561968 Ki > 4000 nM T00663 CO9KP5 11583459 IC50 > 10000 nM T00663 CMIL86 11590363 Ki = 61 nM T00663 C5B3XJ 11620410 IC50 > 40000 nM T00663 CHB3F2 11626055 IC50 = 572 nM T00663 CGX96V 11626927 IC50 < 15848.93 nM T00663 C9T6SC 11640926 Ki = 18 nM T00663 C9VP4Y 11655237 IC50 = 82 nM T00663 CJ9KN7 11683817 IC50 > 10000 nM T00663 CU0E8O 11690457 Ki > 4000 nM T00663 CB0AP2 11705863 Ki > 4000 nM T00663 CVX17E 11740117 IC50 = 32 nM T00663 CS36BH 11843159 IC50 > 5000 nM T00663 CBC08P 11846124 IC50 = 60 nM T00663 CD60CH 11846125 IC50 = 37 nM T00663 CAZS08 11848309 IC50 > 10000 nM T00663 C43IVN 11848567 IC50 > 10000 nM T00663 C9LAY8 11848825 IC50 > 10000 nM T00663 CC09DE 11955790 IC50 = 59 nM T00663 CIQ7M6 14198571 IC50 > 15848.93 nM T00663 CH19QA 15680125 IC50 > 15848.93 nM T00663 CBF4X2 15991561 IC50 = 3162.28 nM T00663 C8TW5P 16007071 IC50 = 2.5 nM T00663 CFPW41 16007116 IC50 = 120 nM T00663 C9TU1O 16046126 IC50 > 1000 nM T00663 CKR57M 16086104 IC50 > 5000 nM T00663 C16NRY 16086114 IC50 = 145 nM T00663 C7Z4LV 16095343 IC50 > 10000 nM T00663 CQG45C 16109001 IC50 = 40000 nM T00663 CK1SZ0 16115350 IC50 > 10000 nM T00663 CZL8G5 16115351 IC50 = 540 nM T00663 CRO0D5 16115352 IC50 = 3500 nM T00663 C0C5AZ 16129582 IC50 = 57 nM T00663 CU56EW 16664858 IC50 = 251.19 nM T00663 C0PS7U 16750106 IC50 = 150 nM T00663 C5IYQ1 17027307 IC50 = 810 nM T00663 CL9BQ6 17748275 IC50 = 40000 nM T00663 C4SPG1 19007057 Ki > 4000 nM T00663 CC1E7R 21078798 Ki > 4000 nM T00663 C95ORH 22261071 IC50 = 52 nM T00663 CE7K3W 23532567 IC50 > 10000 nM T00663 CR3M1N 23644582 Ki > 4000 nM T00663 CVOT06 24535122 IC50 = 6900 nM T00663 CV9U8E 24745781 IC50 > 10000 nM T00663 C9FJZ6 24779711 IC50 = 120 nM T00663 CIN29Y 24801862 IC50 = 3 nM T00663 CZ12SD 24801863 IC50 = 270 nM T00663 C16DKC 24810995 IC50 > 300 nM T00663 CC8Y1U 24810996 IC50 = 360 nM T00663 CH21WG 24810997 IC50 = 96 nM T00663 CQ1D8M 24810999 IC50 = 360 nM T00663 CNI4W8 24811099 IC50 = 680 nM T00663 C0MXK3 24811100 IC50 = 260 nM T00663 CFZN51 24811101 IC50 = 110 nM T00663 CRF71M 24811102 IC50 = 50 nM T00663 CB8A2T 24811103 IC50 > 10000 nM T00663 CJ7M8K 24823663 IC50 = 114 nM T00663 CX0S9L 24854902 IC50 = 9487 nM T00663 C1SVT2 24854903 IC50 > 10000 nM T00663 C61KPI 24856363 IC50 > 16000 nM T00663 C4OWF8 24875373 IC50 = 85 nM T00663 CY8L7E 24896769 IC50 > 10000 nM T00663 C8DG1Y 24941253 IC50 = 6626 nM T00663 C6CVK4 24959046 IC50 > 100000 nM T00663 CU7I2E 24963046 IC50 = 788 nM T00663 CS3Q8B 24995659 Ki > 4000 nM T00663 CD0TB3 25024184 IC50 = 129 nM T00663 C6NU1D 25071599 IC50 = 325 nM T00663 CXD9K3 25071600 IC50 = 61 nM T00663 CYJ8F1 25074077 IC50 = 1000 nM T00663 C4OA5D 25113170 IC50 = 100 nM T00663 CF7C5B 25129829 IC50 > 10000 nM T00663 CXNM84 25129830 IC50 > 10000 nM T00663 CY2S1P 25129831 IC50 > 10000 nM T00663 CCK8D2 25154767 IC50 > 20000 nM T00663 C9ZKH4 25174103 IC50 = 9 nM T00663 CPY2C9 25203945 IC50 = 398.11 nM T00663 CEFT59 25210489 IC50 = 330 nM T00663 CXE16F 25218564 IC50 = 5011 nM T00663 C3RH2Q 25218565 IC50 = 6310 nM T00663 CMF51N 25222038 IC50 = 148 nM T00663 C15DIA 25222587 IC50 = 79 nM T00663 C7BAN0 25262260 IC50 > 20000 nM T00663 CV7AG6 25660569 IC50 = 1500 nM T00663 C5GZ8L 26704995 IC50 = 3900 nM T00663 CRY5L4 42537838 IC50 = 1200 nM T00663 CWS37O 42618140 IC50 > 25118.86 nM T00663 C2JV3O 42618143 IC50 > 25118.86 nM T00663 CG01BO 42618144 IC50 > 25118.86 nM T00663 CI5AE0 43623574 IC50 = 17200 nM T00663 C0HB4C 44129168 IC50 = 16800 nM T00663 CX16AN 44138038 Ki = 16 nM T00663 CO42DC 44138048 IC50 = 316.23 nM T00663 CL65QV 44138049 IC50 = 125.89 nM T00663 CR7TY6 44197572 IC50 > 20000 nM T00663 C1G2ZQ 44198874 IC50 > 20000 nM T00663 C75TAQ 44200209 IC50 = 83 nM T00663 C7W4AX 44200211 IC50 = 320 nM T00663 C16HSY 44200344 IC50 = 68 nM T00663 CBY7T8 44200468 IC50 = 510 nM T00663 C8KNA3 44219632 Ki > 4000 nM T00663 C0VIX4 44219633 Ki > 4000 nM T00663 CPT6F0 44224261 IC50 = 160 nM T00663 CMRG01 44236943 IC50 = 9900 nM T00663 C0HM6Z 44236944 IC50 = 900 nM T00663 CRT04D 44236945 IC50 = 2200 nM T00663 C46EDI 44236946 IC50 = 540 nM T00663 C37IRD 44236947 IC50 = 960 nM T00663 CGSA21 44236948 IC50 = 250 nM T00663 CGO6L3 44236949 IC50 = 1100 nM T00663 CYV31G 44236950 IC50 = 1400 nM T00663 C2D4LE 44236951 IC50 = 1000 nM T00663 C6IGK2 44236952 IC50 > 20000 nM T00663 CFU45N 44236953 IC50 > 20000 nM T00663 C07YUQ 44236954 IC50 = 200 nM T00663 C8HPQ7 44236955 IC50 = 290 nM T00663 CG8KU3 44236956 IC50 > 20000 nM T00663 CLK0U1 44236957 IC50 > 20000 nM T00663 C9L3XK 44236958 IC50 > 20000 nM T00663 CRJ9F0 44236959 IC50 > 20000 nM T00663 CBXL42 44236960 IC50 = 310 nM T00663 C9HR2S 44236961 IC50 = 1800 nM T00663 C1CD6L 44236962 IC50 = 2300 nM T00663 C34TLE 44236963 IC50 = 5000 nM T00663 CW3PO4 44236964 IC50 = 8900 nM T00663 CC93MW 44236965 IC50 = 5800 nM T00663 C1XQG3 44236966 IC50 = 2000 nM T00663 C82AFZ 44236967 IC50 = 2000 nM T00663 CTH0D7 44236968 IC50 = 6400 nM T00663 COF30J 44236969 IC50 > 20000 nM T00663 C6J0UF 44236970 IC50 > 20000 nM T00663 CP81MF 44236971 IC50 = 60 nM T00663 CTHS64 44236972 IC50 = 80 nM T00663 CNL6H4 44236973 IC50 = 410 nM T00663 C87WNK 44236974 IC50 = 210 nM T00663 CJ9VI7 44236975 IC50 = 530 nM T00663 C0FT5H 44236976 IC50 = 350 nM T00663 C1HX8I 44236977 IC50 = 1000 nM T00663 CET82Q 44236978 IC50 = 110 nM T00663 C59YJV 44236979 IC50 = 4800 nM T00663 CSI8C1 44236980 IC50 = 620 nM T00663 CF2YU6 44236981 IC50 = 11000 nM T00663 C19NBZ 44236982 IC50 > 20000 nM T00663 CH56RI 44404432 IC50 = 270 nM T00663 CUW89Z 44404434 IC50 = 10.9 nM T00663 CW8F3T 44404438 IC50 = 233 nM T00663 C9AJ1Y 44404441 IC50 = 3 nM T00663 C2RXS6 44404444 IC50 = 130 nM T00663 C2MT9X 44404797 IC50 = 3.3 nM T00663 CAC7Q5 44404813 IC50 = 1.259 nM T00663 C7F6KQ 44408641 IC50 = 8 nM T00663 C27KEP 44408669 IC50 = 44 nM T00663 CFY5E9 44408670 IC50 = 6 nM T00663 CI76KB 44408825 IC50 = 9 nM T00663 C3I1VN 44408826 IC50 = 207 nM T00663 CBC3X6 44408908 IC50 = 5 nM T00663 CY8LJ5 44408909 IC50 = 10 nM T00663 C3O7GC 44408936 IC50 = 15 nM T00663 CCW09A 44408944 IC50 = 3 nM T00663 C5YUK6 44431823 IC50 = 630.96 nM T00663 CO91FC 44431824 IC50 = 1000 nM T00663 CI95TS 44431825 IC50 > 15848.93 nM T00663 CJN16A 44431826 IC50 > 15848.93 nM T00663 CU75OI 44431827 IC50 > 15848.93 nM T00663 C2P8TK 44431828 IC50 > 15848.93 nM T00663 C2C4SX 44431829 IC50 = 2511.89 nM T00663 C9Y1ID 44431830 IC50 = 3162.28 nM T00663 CU20ER 44431831 IC50 = 251.19 nM T00663 CL87AX 44431832 IC50 = 1000 nM T00663 CA61VJ 44431833 IC50 = 501.19 nM T00663 C1KW0V 44431834 IC50 = 1584.89 nM T00663 CAX8F5 44440161 IC50 = 412 nM T00663 CM2E3N 44440217 IC50 = 708 nM T00663 C6RD3G 44440219 IC50 = 582 nM T00663 CIAJ70 44440220 IC50 = 5000 nM T00663 C52CDB 44440221 IC50 = 32 nM T00663 CFZS24 44440223 IC50 = 107 nM T00663 CSA87R 44440224 IC50 = 31 nM T00663 CH76CV 44440225 IC50 = 14 nM T00663 CKSO82 44440228 IC50 = 179 nM T00663 C8HWI1 44440229 IC50 = 120 nM T00663 CVD97U 44440230 IC50 = 48 nM T00663 C9AV4C 44440236 IC50 = 5 nM T00663 C60YEU 44444010 IC50 = 1000 nM T00663 C1HEB4 44444011 IC50 > 20000 nM T00663 CKB97N 44444012 IC50 = 3600 nM T00663 CE02WM 44444013 IC50 = 1300 nM T00663 C7GFW0 44444014 IC50 = 510 nM T00663 CZ73CR 44444016 IC50 = 1600 nM T00663 C7FTV8 44444018 IC50 = 530 nM T00663 C52NJF 44444019 IC50 = 930 nM T00663 CY0G7R 44444021 IC50 = 210 nM T00663 C5I8ND 44444024 IC50 = 440 nM T00663 CA7N3G 44444025 IC50 = 480 nM T00663 C0JGC3 44444026 IC50 = 3600 nM T00663 CER95H 44444027 IC50 = 760 nM T00663 C16XZW 44444028 IC50 = 15000 nM T00663 CA8Q2M 44444029 IC50 = 6500 nM T00663 CL4B1D 44444030 IC50 = 140 nM T00663 CAX59T 44444031 IC50 = 490 nM T00663 C0CIN7 44444033 IC50 > 20000 nM T00663 CY20IT 44444034 IC50 = 5200 nM T00663 CKD8E0 44444036 IC50 = 5000 nM T00663 CD8BK3 44444037 IC50 = 250 nM T00663 CDZO02 44444038 IC50 = 200 nM T00663 C7H3AL 44444039 IC50 = 240 nM T00663 CXK91I 44444991 IC50 = 7 nM T00663 CCP02M 44444992 IC50 = 3 nM T00663 CU80BP 44517743 IC50 > 10000 nM T00663 CKV96M 44571730 IC50 > 20000 nM T00663 C7Q1VU 44580077 IC50 > 16000 nM T00663 CL90SE 44580358 IC50 > 16000 nM T00663 CK1VE7 44580420 IC50 > 16000 nM T00663 CH2R7X 44580449 IC50 > 16000 nM T00663 C1VH0C 44580532 IC50 > 16000 nM T00663 CXC52J 44580649 IC50 > 16000 nM T00663 CE32BQ 44580689 IC50 > 16000 nM T00663 C8Z5AX 44580778 IC50 > 16000 nM T00663 C5Z3LI 44591740 IC50 = 16 nM T00663 CZ8XI5 44627578 Ki = 130 nM T00663 CKM3N2 44627579 IC50 = 297 nM T00663 CN30CM 44627580 IC50 = 365 nM T00663 C7NU3G 44627581 IC50 = 7 nM T00663 CDF41Q 44627582 IC50 = 4 nM T00663 CKI17J 44627583 IC50 = 390 nM T00663 C7EK0M 44627681 IC50 = 79 nM T00663 C8RVP9 44627682 IC50 = 140 nM T00663 C6E2LI 44627683 IC50 = 85 nM T00663 C21IGV 44627684 IC50 = 133 nM T00663 CG6UW5 44634494 IC50 = 13760 nM T00663 CJ0LU4 45104966 IC50 = 263 nM T00663 CJ32SA 45203151 IC50 = 1100 nM T00663 C2JVA4 45270368 IC50 = 250 nM T00663 CA4XQ3 45375859 IC50 = 5456 nM T00663 C46MWH 45488127 IC50 = 3950 nM T00663 C3P8YT 45488146 IC50 = 31800 nM T00663 CW2G7D 46868853 IC50 = 7 nM T00663 CR57OZ 46868855 IC50 = 324 nM T00663 CI8YE5 46868856 IC50 = 12 nM T00663 C94EPL 46868925 IC50 = 5 nM T00663 C0GU4D 46868930 IC50 = 160 nM T00663 C9ULP0 46869071 IC50 = 5300 nM T00663 CU52JS 46869075 IC50 = 3600 nM T00663 CFQT10 46869147 IC50 = 42500 nM T00663 CEK2I5 46869149 IC50 = 820 nM T00663 C2XQ4K 46869223 IC50 = 9400 nM T00663 C8U1AH 46869285 IC50 = 6 nM T00663 CKTD23 46869290 IC50 = 183 nM T00663 CV57OI 46869490 IC50 = 9 nM T00663 C9XHK0 46869491 IC50 = 14 nM T00663 C47JSD 46869493 IC50 = 14 nM T00663 C65NDB 46869609 IC50 = 31500 nM T00663 CP2A4Y 46869611 IC50 = 550 nM T00663 CQ0AU8 46869671 IC50 = 45600 nM T00663 C4RS7M 46869672 IC50 = 465 nM T00663 C1VZM6 46869673 IC50 = 5 nM T00663 CYI69K 46869674 IC50 = 25 nM T00663 C2PC6T 46869677 IC50 = 1500 nM T00663 CSL2N6 46869740 IC50 = 5900 nM T00663 C6V9CD 46869741 IC50 = 25 nM T00663 CZCQ05 46869742 IC50 = 1600 nM T00663 C09GAW 46869745 IC50 = 143 nM T00663 CVBG98 46869815 IC50 = 594 nM T00663 CU2D5N 46869816 IC50 = 18 nM T00663 C8WH7Q 46869817 IC50 = 80 nM T00663 CFOX43 46869876 IC50 = 197 nM T00663 CE0CY1 46869877 IC50 = 560 nM T00663 C2DW6T 46869878 IC50 = 33 nM T00663 C19DQG 46869879 IC50 = 34 nM T00663 CR1OH0 46869880 IC50 = 6 nM T00663 C8SFI1 46869881 IC50 = 9 nM T00663 CD1YH9 46869882 IC50 = 28 nM T00663 CQIC19 46879806 IC50 > 20000 nM T00663 C6WD4Q 46881329 IC50 = 6309.57 nM T00663 C6GQH3 46881341 IC50 = 12589.25 nM T00663 CEK6A9 46881342 IC50 = 3981.07 nM T00663 C84TWY 46881343 IC50 > 15848.93 nM T00663 C1DFI0 46881344 IC50 = 5011.87 nM T00663 CW32UX 46881345 IC50 > 15848.93 nM T00663 C8CE7P 46881351 IC50 = 10000 nM T00663 C7AE4V 46881352 IC50 = 1000 nM T00663 CP7UE5 46881353 IC50 > 15848.93 nM T00663 C32XZI 46881354 IC50 = 15848.93 nM T00663 CSQ8O9 46881355 IC50 = 6309.57 nM T00663 CO0SC4 46881358 IC50 = 1995.26 nM T00663 C4DXW0 46881359 IC50 = 630.96 nM T00663 CK67BQ 46881360 IC50 > 15848.93 nM T00663 CV4O5T 46881361 IC50 > 15848.93 nM T00663 CRD8S3 46884198 IC50 = 10.9 nM T00663 CRKV43 46884199 Ki = 5 nM T00663 CA2Y8J 46901260 IC50 > 20000 nM T00663 CQR9K1 46933384 IC50 > 100000 nM T00663 CHSF07 49806372 IC50 > 1000 nM T00663 CS18HZ 49839481 IC50 = 77 nM T00663 C83VHI 49864785 IC50 = 90000 nM T00663 C2UTK6 49864850 IC50 > 100000 nM T00663 CAE53W 49865153 IC50 = 78000 nM T00663 CDR47S 49867175 IC50 = 25 nM T00663 CH4FY5 50941455 IC50 = 24 nM T00663 CBR71Y 50941538 IC50 = 16 nM T00663 C4BN7W 50941539 IC50 = 29 nM T00663 C1HI2W 51346940 IC50 = 40 nM T00663 C5GPU9 51346941 IC50 = 90 nM T00663 CM24LF 52938983 IC50 > 20000 nM T00663 CA7HQ9 52941011 IC50 = 700 nM T00663 CA6BH5 52941226 IC50 = 5400 nM T00663 CMXC68 52941286 IC50 = 1500 nM T00663 C0DSA8 52941649 IC50 = 17000 nM T00663 C4O3RZ 52942227 IC50 > 50000 nM T00663 C3BKR7 52942436 IC50 = 6500 nM T00663 C8R9SA 52942482 IC50 = 37000 nM T00663 CAC3J5 52942507 IC50 = 1600 nM T00663 CTPH98 52942532 IC50 > 50000 nM T00663 CHP7M6 52943427 IC50 > 50000 nM T00663 CS8VA0 52943431 IC50 = 4400 nM T00663 CJU79I 52943626 IC50 = 900 nM T00663 C07JYV 52944873 IC50 = 2100 nM T00663 CB1UJ7 52944909 IC50 = 1600 nM T00663 CD2WZ5 52944914 IC50 = 1600 nM T00663 CY9B7D 52944962 IC50 > 50000 nM T00663 C1Z7KR 52946059 IC50 = 9000 nM T00663 CCMX82 52946092 IC50 = 27000 nM T00663 CPIK13 52946145 IC50 = 12600 nM T00663 C67TBV 52946152 IC50 = 1400 nM T00663 C6OH8X 52946172 IC50 > 50000 nM T00663 CC6Z1J 52947386 IC50 = 3800 nM T00663 CC5P4R 52947399 IC50 > 50000 nM T00663 C9O7FN 52947421 IC50 > 50000 nM T00663 C72TPI 52947422 IC50 > 50000 nM T00663 C3R4FI 52948519 IC50 = 920 nM T00663 CLU92X 52948565 IC50 = 31000 nM T00663 CDXL70 52948593 IC50 = 470 nM T00663 CO3EL9 52948602 IC50 > 50000 nM T00663 C3WHA1 52949737 IC50 > 50000 nM T00663 CMT75N 52949817 IC50 = 610 nM T00663 CBAD62 52949818 IC50 = 610 nM T00663 CSOB70 52950113 IC50 = 690 nM T00663 CW2KE5 53317337 IC50 = 38800 nM T00663 CJQN83 53317338 IC50 = 3020 nM T00663 CJ2P3V 53317339 IC50 = 504 nM T00663 C9E3FV 53317340 IC50 = 226 nM T00663 CBTX53 53317412 IC50 = 16000 nM T00663 COCN94 53317413 IC50 = 40 nM T00663 CHC29T 53317414 IC50 = 210 nM T00663 C82LCE 53317415 IC50 = 590 nM T00663 CR0DJ1 53317416 IC50 = 92 nM T00663 C28JAP 53317417 IC50 = 36 nM T00663 C8Q0OR 53318506 IC50 = 62 nM T00663 CP7T3N 53318709 IC50 = 54 nM T00663 CKD47I 53319944 IC50 = 99 nM T00663 CP7BR1 53319945 IC50 = 1020 nM T00663 C3TAC2 53320021 IC50 = 3900 nM T00663 COPI53 53321333 IC50 = 410 nM T00663 C0GLS5 53321334 IC50 = 120 nM T00663 C2V0QU 53321577 IC50 = 250 nM T00663 CG8KC9 53322569 IC50 = 9110 nM T00663 C3SA1K 53322570 IC50 = 310 nM T00663 COG9J2 53322644 IC50 = 130 nM T00663 CUR1A6 53322645 IC50 = 70 nM T00663 C25OEY 53322984 IC50 = 125 nM T00663 CK8Y5F 53323911 IC50 = 162 nM T00663 C9SHJ0 53323985 IC50 = 85 nM T00663 C49MDG 53323986 IC50 = 70 nM T00663 C3AVG0 53323987 IC50 = 430 nM T00663 C18SCR 53323988 IC50 = 14 nM T00663 C38RXW 53323989 IC50 = 22 nM T00663 CXWB94 53325188 IC50 = 110 nM T00663 C8VPW5 53325283 IC50 = 54 nM T00663 CA3X2Q 53325284 IC50 = 130 nM T00663 CIG7X9 53325285 IC50 = 94 nM T00663 C4A8JK 53325286 IC50 = 100 nM T00663 CI1RT4 53325287 IC50 = 280 nM T00663 CNT50E 53325288 IC50 = 24 nM T00663 CR91NJ 53325555 IC50 = 700 nM T00663 CBW0G7 53326484 IC50 = 9620 nM T00663 CV7I4O 53326555 IC50 = 32 nM T00663 C27IBZ 53326556 IC50 = 61 nM T00663 C5UK3J 53326557 IC50 = 950 nM T00663 CVJ6K9 53326558 IC50 = 160 nM T00663 C8NA4L 53384644 IC50 > 30000 nM T00663 CD0ZI6 53469858 IC50 = 245 nM T00663 CCG3H2 54580285 IC50 = 10 nM T00663 CJDM48 54580615 IC50 = 600 nM T00663 CPRC42 54580619 IC50 = 160 nM T00663 C56ARZ 54580647 IC50 = 7 nM T00663 CB4TJ8 54581287 IC50 = 50 nM T00663 C5U6YP 54581288 IC50 = 700 nM T00663 CNU9G4 54581289 IC50 = 4400 nM T00663 C39VAB 54581290 IC50 = 210 nM T00663 CT3JS6 54581291 IC50 = 7 nM T00663 CM7H3P 54581292 IC50 = 9 nM T00663 CEP18Y 54581359 IC50 > 50000 nM T00663 C6JPE1 54581360 IC50 = 52.2 nM T00663 CD2YU5 54581361 IC50 = 4480 nM T00663 C49RNQ 54581362 IC50 = 1230 nM T00663 CA8U3P 54581363 IC50 > 50000 nM T00663 C2ZN7A 54581623 IC50 = 1450 nM T00663 CH6VE9 54581624 IC50 = 160 nM T00663 CD4Z6Y 54581656 IC50 = 1330 nM T00663 C5V6OY 54582175 IC50 > 30000 nM T00663 C6B2UL 54582304 IC50 = 63 nM T00663 C1FR4Q 54582305 IC50 = 20 nM T00663 CP4HV1 54582306 IC50 = 10 nM T00663 CFG68S 54582307 IC50 = 4 nM T00663 C52OMN 54582618 IC50 = 340 nM T00663 C26UOY 54582645 IC50 = 240 nM T00663 C1OM6E 54583278 IC50 = 20 nM T00663 CNE41S 54583279 IC50 = 90 nM T00663 C6XC0E 54583280 IC50 = 30 nM T00663 CMCL04 54583281 IC50 = 60 nM T00663 CTQ70F 54583282 IC50 = 50 nM T00663 CCO5I2 54583368 IC50 = 12600 nM T00663 CECO89 54583369 IC50 = 1910 nM T00663 CFV81A 54583573 IC50 = 70 nM T00663 C0K8HF 54583574 IC50 = 200 nM T00663 CS83TL 54583576 IC50 = 320 nM T00663 CF72GE 54583602 IC50 = 390 nM T00663 C68FYO 54583603 IC50 = 1400 nM T00663 CM1TU0 54584242 IC50 = 70 nM T00663 CP6K3I 54584243 IC50 = 60 nM T00663 CR4E7O 54584244 IC50 = 80 nM T00663 CRKI30 54584315 IC50 = 945 nM T00663 C3P2HM 54584316 IC50 = 30400 nM T00663 CL69AG 54584317 IC50 = 364 nM T00663 CBA65Z 54584562 IC50 = 730 nM T00663 C2DRY7 54584563 IC50 = 130 nM T00663 C7GR5M 54584564 IC50 = 160 nM T00663 CC3BE2 54584594 IC50 = 650 nM T00663 CEJ0M6 54584595 IC50 = 340 nM T00663 C3EP6K 54584596 IC50 = 110 nM T00663 CD4WJ7 54584597 IC50 = 400 nM T00663 CT16HO 54585212 IC50 = 30 nM T00663 CNB2M9 54585213 IC50 = 90 nM T00663 CC8YN2 54585285 IC50 = 14800 nM T00663 CGA8X9 54585286 IC50 > 50000 nM T00663 CV69FU 54585287 IC50 > 50000 nM T00663 CR1X8Y 54585288 IC50 = 1030 nM T00663 CTY84H 54585289 IC50 > 50000 nM T00663 CWE79L 54585290 IC50 = 4810 nM T00663 C0FAG2 54585291 IC50 = 2460 nM T00663 CNLU49 54585292 IC50 = 4130 nM T00663 CPZ20X 54585507 IC50 = 100 nM T00663 CNUP53 54586040 IC50 = 880 nM T00663 C30VTY 54586163 IC50 = 170 nM T00663 CQNZ54 54586164 IC50 = 190 nM T00663 CUD8J0 54586233 IC50 = 49100 nM T00663 CT78AW 54586474 IC50 = 860 nM T00663 CGW36K 54586475 IC50 = 160 nM T00663 CE0C3W 54586476 IC50 = 200 nM T00663 C8IO1D 54586477 IC50 = 480 nM T00663 CWX92H 54586479 IC50 = 170 nM T00663 C40EQC 54586508 IC50 = 390 nM T00663 C6BX0V 54587174 IC50 = 730 nM T00663 CI49LN 54587175 IC50 > 20000 nM T00663 CI8ZH6 54587176 IC50 = 50 nM T00663 C1V8HM 54587177 IC50 = 60 nM T00663 CO1JB2 54587178 IC50 = 20 nM T00663 C3JAW8 54587179 IC50 = 30 nM T00663 CA5N6I 54587258 IC50 = 27400 nM T00663 CKX15Q 54587259 IC50 = 18300 nM T00663 CKQS27 54587260 IC50 = 14900 nM T00663 C57LBW 54587261 IC50 = 2670 nM T00663 CMH8N5 54587504 IC50 = 630 nM T00663 C8UC1Z 54587510 IC50 = 750 nM T00663 CL75DP 54587542 IC50 = 150 nM T00663 C0I4FV 54764508 IC50 = 37 nM T00663 C18TKF 54764593 IC50 = 7 nM T00663 CG78UW 56658171 IC50 = 11 nM T00663 C7LDZ3 56658303 IC50 = 280 nM T00663 C0MW6D 56658304 IC50 = 8 nM T00663 CK18JP 56661802 IC50 = 41 nM T00663 CE1O3B 56661803 IC50 = 14 nM T00663 CSJ6A9 56665092 IC50 = 3 nM T00663 C7HA6J 56665093 IC50 = 8 nM T00663 CS5HP6 56665245 IC50 = 30 nM T00663 C4SO3M 56665246 IC50 = 6 nM T00663 CE2PY0 56665247 IC50 = 6 nM T00663 C9AW1E 56668539 IC50 = 15 nM T00663 C0MR6D 56668696 IC50 = 7 nM T00663 CXF3R9 56668697 IC50 = 19 nM T00663 CU3I2J 56672173 IC50 = 71 nM T00663 CJ9I6K 56672174 IC50 = 2 nM T00663 CD5NZ4 56672175 IC50 = 6 nM T00663 CRAK61 56675421 IC50 = 8 nM T00663 CG3ZU0 56678888 IC50 = 52 nM T00663 CAP1M2 56682209 IC50 = 24 nM T00663 C9DO8G 56682210 IC50 = 2 nM T00663 CTO6N5 56834943 IC50 = 24 nM T00663 C97SLT 57340680 IC50 = 704 nM T00663 C0UDN5 57340685 IC50 = 130 nM T00663 CDP45J 57390517 IC50 = 140 nM T00663 C28LIB 57390518 IC50 = 130 nM T00663 C8DZ1N 57390519 IC50 = 12 nM T00663 C7K4LJ 57390520 IC50 = 240 nM T00663 C32DFY 57390767 IC50 = 140 nM T00663 CKUX48 57390768 IC50 = 200 nM T00663 C32FUN 57390769 IC50 = 72 nM T00663 C6P0YR 57390770 IC50 = 17 nM T00663 CH4X7D 57390771 IC50 = 160 nM T00663 CG51FX 57392289 IC50 = 31 nM T00663 C9EJN6 57392581 IC50 = 380 nM T00663 CP1D7N 57392582 IC50 = 320 nM T00663 CX0F1Z 57392583 IC50 = 78 nM T00663 C2IZ3W 57392739 IC50 = 7 nM T00663 C9P1SC 57393560 IC50 = 16 nM T00663 CVH4X0 57394043 IC50 = 17 nM T00663 CN3MB5 57394305 IC50 = 100 nM T00663 CLOD68 57394306 IC50 = 34 nM T00663 C1EYU6 57394468 IC50 = 32 nM T00663 CV9W8C 57395293 IC50 = 24 nM T00663 CQ2A1B 57395802 IC50 = 63 nM T00663 C15YOZ 57396060 IC50 = 48 nM T00663 CL4BN7 57396061 IC50 = 110 nM T00663 CW7XA9 57397040 IC50 = 13 nM T00663 C18MFO 57397857 IC50 = 35 nM T00663 C7KJ2W 57397858 IC50 = 2200 nM T00663 CB7DO2 57397859 IC50 = 49 nM T00663 CDI28Y 57397860 IC50 = 60 nM T00663 CKG0P1 57397861 IC50 = 170 nM T00663 C9A7RL 57397862 IC50 = 140 nM T00663 CH1QI7 57399519 IC50 = 27 nM T00663 CA0SR3 57399520 IC50 = 200 nM T00663 C8IFD4 57399521 IC50 = 48 nM T00663 CT5S8H 57400156 IC50 = 100 nM T00663 C2DG7X 57401275 IC50 = 45 nM T00663 C8FQH3 57402785 IC50 > 1000 nM T00663 C1HD8L 57402972 IC50 = 520 nM T00663 C8ZQ3A 57403022 IC50 = 70 nM T00663 CKIX12 57403023 IC50 = 15 nM T00663 C4VKU7 57403024 IC50 = 70 nM T00663 CZ5L4E 57403025 IC50 = 3500 nM T00663 CNP8C3 57403026 IC50 = 990 nM T00663 CDXK85 57403027 IC50 = 80 nM T00663 CH0NB1 57403028 IC50 = 2200 nM T00663 CJY46H 57403029 IC50 = 30 nM T00663 CI1A8M 57404048 IC50 = 7738 nM T00663 C6UAN1 57467725 IC50 = 2199 nM T00663 C7I4QD 57519510 IC50 = 159 nM T00663 CO57NK 58155042 IC50 = 680 nM T00663 CT3EW2 59292007 IC50 = 560 nM T00663 COH62U 60097413 IC50 > 3300 nM T00663 C06UMH 66958119 IC50 = 326 nM T00663 CV63UL 67240318 IC50 > 10000 nM T00663 C69OHY 68560854 IC50 > 20000 nM T00663 C25MEI 68561431 IC50 > 20000 nM T00663 CCD89X 68563058 IC50 > 20000 nM T00663 C0XCY9 68565200 IC50 > 20000 nM T00663 CW6BH7 68566254 IC50 > 20000 nM T00663 CQRP72 68567556 IC50 > 20000 nM T00663 C48EIQ 68568011 IC50 > 20000 nM T00663 CAWC35 68621678 IC50 > 1000 nM T00663 C3GTU1 69762142 IC50 > 10000 nM T00663 CQ8HE2 70690944 IC50 > 30000 nM T00663 C13FWG 70695135 IC50 > 30000 nM T00663 C0VZB2 70697173 IC50 > 30000 nM T00663 C2LU7I 70702008 IC50 = 7 nM T00663 CMPK41 70702010 IC50 = 117 nM T00663 CKT98U 71584212 IC50 = 1090 nM T00663 CI3MH6 71602620 IC50 > 20000 nM T00663 CCD0W3 71602669 IC50 = 24 nM T00663 C3D1CA 71602671 IC50 = 33 nM T00663 CG1DR3 71602672 IC50 = 12 nM T00663 CQ9A6D 71602719 IC50 = 46 nM T00663 CDU4I0 71602720 IC50 = 59 nM T00663 CP01YB 71602721 IC50 = 32 nM T00663 CX60NJ 71602722 IC50 = 38 nM T00663 CHU36E 71602723 IC50 = 54 nM T00663 C7MGB8 71602768 IC50 = 77 nM T00663 CZ8US1 71602769 IC50 = 43 nM T00663 C2GM5W 71602770 IC50 = 22 nM T00663 C9UY4L 71602771 IC50 = 15 nM T00663 C6O2KE 71602772 IC50 = 120 nM T00663 CA2J9W 71602817 IC50 = 250 nM T00663 CS4K2F 71602818 IC50 = 35 nM T00663 CY8H5Z 71602819 IC50 = 1400 nM T00663 C60VBS 71602820 IC50 = 63 nM T00663 CI09ER 71602821 IC50 = 50 nM T00663 C2KW8Y 71602864 IC50 = 640 nM T00663 CEX14A 71602865 IC50 = 640 nM T00663 CEF41S 71602866 IC50 = 110 nM T00663 CAM32B 71602867 IC50 = 120 nM T00663 CDH23B 71602868 IC50 = 80 nM T00663 CVUG79 71602911 IC50 = 170 nM T00663 C8AM1K 71655603 IC50 > 20000 nM T00663 C7OQC1 71720177 IC50 = 1860 nM T00663 CD3JF9 71745086 IC50 = 40 nM T00663 CZ4BX1 72547959 IC50 = 364 nM T00663 C8THP4 72946274 IC50 = 26 nM T00663 CYZP14 72946275 IC50 > 20000 nM T00663 C8T2WZ 72946276 IC50 = 70 nM T00663 C5N9JK 72946277 IC50 = 32 nM T00663 C3TM0X 72946450 IC50 = 126 nM T00663 CP8ZR3 72946451 IC50 = 523 nM T00663 C1IKA3 72946452 IC50 = 366 nM T00663 CWG15I 72946453 IC50 = 27 nM T00663 C2I8CL 72946454 IC50 = 134 nM T00663 CV5P7N 72946655 IC50 = 216 nM T00663 C98FIU 72946656 IC50 = 1 nM T00663 CJA75F 72946661 IC50 = 435 nM T00663 C0QL7V 72946851 IC50 = 19 nM T00663 C8GI2A 72946852 IC50 = 74 nM T00663 C1NKW5 72946853 IC50 = 52 nM T00663 C78GOJ 72946854 IC50 = 16 nM T00663 CO61VP 72946855 IC50 = 187 nM T00663 CG4YH2 72946856 IC50 = 24 nM T00663 C0HQ6V 72947058 IC50 = 587 nM T00663 C8J3WG 76328237 IC50 = 7 nM T00663 CJ2T9E 76332983 IC50 > 10000 nM T00663 CLTG58 78350466 IC50 = 1600 nM T00663 C54KDR 86763302 IC50 = 1895 nM T00663 C4HKT5 87057579 IC50 = 98 nM T00663 CQ2OB9 90292687 IC50 > 10000 nM T00663 CHI39S 90292823 IC50 > 10000 nM T00663 C5C9PB 90667115 IC50 = 218 nM T00663 CI4RH8 90667116 IC50 = 371 nM T00663 C4H0ZN 90667117 IC50 = 414 nM T00663 CTB63D 90667118 IC50 = 727 nM T00663 C5TPF3 90667119 IC50 = 173 nM T00663 C0INK4 90667120 IC50 = 3100 nM T00663 C80FXC 90667121 IC50 = 160 nM T00663 C98QUS 90667122 IC50 > 20000 nM T00663 C4YS9Z 90667123 IC50 = 12000 nM T00663 C4A3FO 90667124 IC50 > 20000 nM T00663 CG6C4H 90667125 IC50 = 132 nM T00663 CQIP37 90667126 IC50 = 374 nM T00663 C0HL7F 90667127 IC50 = 325 nM T00663 C6FRO8 90667128 IC50 = 218 nM T00663 CE0ID8 90667129 IC50 = 371 nM T00663 CZ45HF 90667130 IC50 = 680 nM T00663 CSJ4C2 90667131 IC50 = 326 nM T00663 CJU4V7 90667132 IC50 = 414 nM T00663 CBZ73T 90667133 IC50 = 727 nM T00663 CW3UI2 90667134 IC50 = 173 nM T00663 C0M3VU 90667135 IC50 = 0.28 nM T00663 CH7G1F 90667136 IC50 = 0.42 nM T00663 C7P8TV 90667137 IC50 = 0.78 nM T00663 CE05TI 90667138 IC50 = 0.3 nM T00663 CH4DI3 90667139 IC50 = 0.28 nM T00663 C1U9DY 90667140 IC50 = 0.31 nM T00663 C9JQE0 90667141 IC50 = 0.25 nM T00663 CIV0J1 90667142 IC50 = 1.2 nM T00663 C1C7PW 90667143 IC50 = 0.77 nM T00663 CLF96U 90667144 IC50 = 2.5 nM T00663 C49JZU 90667145 IC50 = 0.16 nM T00663 CE5M7Q 90667146 IC50 = 1800 nM T00663 C7V8BN 91754589 IC50 = 11 nM T00663 CQ2G3S 91754590 IC50 = 15 nM T00663 CJQ5N6 91936970 IC50 = 2100 nM T00663 C2GNI5 101891709 IC50 < 1 nM T00663 C6ZFW9 101913690 IC50 = 18 nM T00663 C9VSP7 101913691 IC50 = 26 nM T00663 C5DLO7 118143962 IC50 = 38 nM T00663 CK7O6G 118144051 IC50 = 230 nM T00663 CQ29IK 118144281 IC50 = 133 nM T00663 CZG4U9 118144359 IC50 = 62 nM T00663 C61FOL 118144367 IC50 = 114 nM T00663 CE7QM9 118144380 IC50 = 169 nM T00663 C8GU6M 118146727 IC50 = 141 nM T00663 CY82JT 118146747 IC50 = 37 nM T00663 CIDU81 118146748 IC50 = 130 nM T00663 C1OIF0 118146749 IC50 > 10000 nM T00663 C8TLS2 118146764 IC50 = 238 nM T00663 C32HVY 118146772 IC50 = 860 nM T00663 CULV52 118146793 IC50 = 71 nM T00663 CB2WI6 118146794 IC50 = 5184 nM T00663 CQFE90 118146797 IC50 = 3063 nM T00663 CA7H9O 118146798 IC50 = 4588 nM T00663 C1MI6J 118146804 IC50 = 23 nM T00663 CERD34 118146805 IC50 = 34 nM T00663 C48AZY 118146813 IC50 = 100 nM T00663 CKT2Q3 118146814 IC50 = 162 nM T00663 CJ4Z3K 118146817 IC50 = 2166 nM T00663 C7Q6RW 118146819 IC50 = 162 nM T00663 CH0I3M 118146826 IC50 = 162 nM T00663 CT29IZ 118146828 IC50 = 203 nM T00663 CHWP46 118146849 IC50 = 313 nM T00663 C4P9AK 118146855 IC50 = 80 nM T00663 CT8K0N 118146868 IC50 = 3300 nM T00663 CET9N4 118146870 IC50 = 31 nM T00663 C4PBE7 118146871 IC50 = 54 nM T00663 C6LEU5 118146872 IC50 = 28 nM T00663 CX08HF 118146873 IC50 = 594 nM T00663 CD8L5Y 118146874 IC50 = 116 nM T00663 CNI34V 118146882 IC50 = 23 nM T00663 C8K0GC 118146884 IC50 = 311 nM T00663 CQW3L7 118146891 IC50 = 201 nM T00663 C4O6MA 118146892 IC50 = 58 nM T00663 CZ35XB 118146932 IC50 = 141 nM T00663 C7NDK6 118146979 IC50 = 21 nM T00663 C56EHT 118146984 IC50 = 139 nM T00663 C3R5DA 118720654 IC50 = 115 nM T00663 C0KM6L 118720655 IC50 = 596 nM T00663 C3FY2J 118720656 IC50 = 1829 nM T00663 CGFD93 118720657 IC50 = 137 nM T00663 C8L9SK 118720658 IC50 = 34 nM T00663 C81HTM 118720659 IC50 = 29 nM T00663 CJ2NI1 118721229 IC50 = 350 nM T00663 CC05EY 118721230 IC50 = 710 nM T00663 C7HJ8Y 118721231 IC50 = 32 nM T00663 C5XMF8 118721232 IC50 = 12 nM T00663 CZY01I 118721233 IC50 = 5.5 nM T00663 C2USQ7 118721234 IC50 = 14 nM T00663 CDS2U3 118721235 IC50 = 31 nM T00663 C0H9OV 118721236 IC50 = 1.9 nM T00663 C83KJY 118721237 IC50 = 1.9 nM T00663 C13QEP 118721238 IC50 = 20 nM T00663 CVC3B0 118721239 IC50 = 7 nM T00663 C2F6MN 118721240 IC50 = 2200 nM T00663 C36PRN 118721241 IC50 = 1200 nM T00663 CY0J8A 118721242 IC50 = 400 nM T00663 CJLX62 118721243 IC50 = 540 nM T00663 C14BFC 118721244 IC50 = 2500 nM T00663 C6ETU2 118721245 IC50 = 400 nM T00663 CC4OF9 118725553 IC50 = 40 nM T00663 CR9ML7 118725554 IC50 = 12 nM T00663 CZ82KA 118725885 IC50 = 4220 nM T00663 CSV5K7 118725886 IC50 = 199 nM T00663 C9XV2B 118725887 IC50 = 1186 nM T00663 C6KCQ9 118725888 IC50 = 266 nM T00663 C6LCD8 118725889 IC50 = 255 nM T00663 CI96GZ 118725890 IC50 = 91 nM T00663 CL3KT6 118725891 IC50 = 269 nM T00663 C2JNF8 118725892 IC50 = 55 nM T00663 CU9KV7 118725893 IC50 = 33 nM T00663 C51HGX 118725894 IC50 = 82 nM T00663 C3HP6G 118725895 IC50 = 47 nM T00663 CR4K1M 118725896 IC50 = 45 nM T00663 C95CUL 118725897 IC50 = 133 nM T00663 CN27BI 118725898 IC50 = 25 nM T00663 CH1VK2 118725899 IC50 = 35 nM T00663 C5IM2Q 118725900 IC50 = 226 nM T00663 CP7DK8 118725901 IC50 = 79 nM T00663 CL8W3Q 118725902 IC50 = 180 nM T00663 CNL1Z4 118725903 IC50 = 2010 nM T00663 C5S2OE 118725904 IC50 = 2633 nM T00663 CL0CJ2 118725905 IC50 = 678 nM T00663 C4UTF5 118725906 IC50 = 2167 nM T00663 C4PQ8K 118725907 IC50 = 1216 nM T00663 CE7ZH9 118725908 IC50 = 170 nM T00663 CM7IQ3 118725909 IC50 = 1528 nM T00663 C3WF5U 118725910 IC50 = 79 nM T00663 CGR19E 118725911 IC50 = 12 nM T00663 CZ8RX6 118725912 IC50 = 61 nM T00663 CU9RB6 118725913 IC50 = 54 nM T00663 CBO8S2 118725914 IC50 = 213 nM T00663 C5CMS9 118725915 IC50 = 17 nM T00663 CEJ7T0 118725916 IC50 = 80 nM T00663 CHT6K9 118728811 Ki > 4000 nM T00663 CUA3Y2 118728812 Ki > 4000 nM T00663 CDQ78G 118728813 Ki > 4000 nM T00663 CZ6XL7 118728814 Ki > 4000 nM T00663 CMO67K 118728815 Ki > 4000 nM T00663 CR2M0Q 118728816 Ki > 4000 nM T00663 C62SCL 118728817 Ki > 4000 nM T00663 CSB30C 118728819 Ki > 4000 nM T00663 CV7XU8 118728820 Ki > 4000 nM T00663 C3J1EX 118728821 Ki > 4000 nM T00663 CIWB78 118728822 Ki > 4000 nM T00663 CP18SE 118728823 Ki > 4000 nM T00663 CM42CA 118728824 Ki > 4000 nM T00663 C9Q7CL 118728825 Ki > 4000 nM T00663 CCR3S0 118728826 Ki > 4000 nM T00663 CH3ZB0 118732094 IC50 > 10000 nM T00663 C0K5LC 118732096 IC50 > 10000 nM T00663 C4HM7F 118732099 IC50 > 10000 nM T00663 C2R9JZ 118732102 IC50 > 10000 nM T00663 C4IQ7C 118732107 IC50 > 10000 nM T00663 CSLU37 118732108 IC50 > 10000 nM T00663 CYRJ23 118732109 IC50 > 10000 nM T00663 CQCX41 118737057 IC50 > 10000 nM T00663 CI6R3E 122178086 IC50 > 10000 nM T00663 CFD0W1 122178087 IC50 > 10000 nM T00663 CRUE70 122178088 IC50 = 532 nM T00663 CMG2E7 122178091 IC50 = 81 nM T00663 CQ0F5Z 122178092 IC50 = 204 nM T00663 C4X7SD 122192466 IC50 > 10000 nM T00663 C0FM1R 130196825 IC50 = 416 nM T00663 C6OXE3 132134663 IC50 >= 1000 nM T00663 CEX92Y 135417092 IC50 = 9760 nM T00663 CRPC85 135432695 IC50 = 8890 nM T00663 CMXR51 135446691 IC50 = 4240 nM T00663 CI1JQ3 135449325 Ki = 550 nM T00663 C8GZ2B 135449326 Ki > 4000 nM T00663 C1JGA6 135454192 IC50 = 2370 nM T00663 CO6I2L 135523935 Ki > 4000 nM T00663 C1Q2AL 135523936 Ki > 4000 nM T00663 C2PQT5 135523937 Ki > 4000 nM T00663 CP2B4U 135523938 Ki > 4000 nM T00663 C0GMF7 135523939 Ki = 840 nM T00663 CSI4D2 135523940 Ki > 4000 nM T00663 COM67B 135523941 Ki = 3100 nM T00663 CX56SF 135523946 Ki = 2800 nM T00663 CWU14F 135523947 Ki = 3300 nM T00663 CX5LG4 135523948 Ki = 3900 nM T00663 CNY53K 135523949 Ki > 4000 nM T00663 C1HUP6 135523950 Ki = 2700 nM T00663 CA7HF8 135523951 Ki = 3000 nM T00663 CT08OB 135523952 Ki = 3400 nM T00663 C28SDI 135523953 Ki > 4000 nM T00663 CJ08EW 135523954 Ki = 1800 nM T00663 CZ87OT 135523955 Ki = 2700 nM T00663 C5Q0GA 135523957 Ki = 790 nM T00663 CF2G9Y 135523958 Ki > 4000 nM T00663 CGHE70 135523959 Ki = 2900 nM T00663 CWZ6R0 135523960 Ki > 4000 nM T00663 CIHM29 135523961 Ki > 4000 nM T00663 CHW83U 135523962 Ki = 3200 nM T00663 CD1G6A 135523963 Ki = 2500 nM T00663 CA41BZ 135523964 Ki = 3100 nM T00663 C4JCM5 135523965 Ki = 2800 nM T00663 C5EYW9 135533810 IC50 = 7650 nM T00663 CPV59N 135685787 Ki > 4000 nM T00663 CM3UC9 135883136 IC50 = 250 nM T00663 CM2UH4 135894362 IC50 > 1000 nM T00663 CY19DW 135894364 IC50 > 1000 nM T00663 CF1PS8 135934877 Ki > 4000 nM T00663 CTRL59 135976660 Ki = 2500 nM T00663 CQ84IZ 136180335 Ki > 4000 nM T00663 CM17FU 136198654 IC50 > 10000 nM T00663 C15HQK 136218656 IC50 > 1000 nM T00663 CZ06UK 136218660 IC50 > 1000 nM T00663 CML48X 136218661 IC50 > 1000 nM T00663 COB69I 136218662 IC50 > 1000 nM T00663 CSL6Q8 136218663 IC50 > 1000 nM T00663 CTFJ83 136226213 IC50 > 1000 nM T00663 C5EV8A 136240902 IC50 > 1000 nM T00663 CX9LB5 136240903 IC50 > 1000 nM T00663 CMC58H 136240944 IC50 > 1000 nM T00663 C60PRZ 136241012 IC50 > 1000 nM T00663 C1Q9YN 136252259 IC50 > 1000 nM T00663 CH9O7Z 137631713 IC50 = 17 nM T00663 C4V1EU 137636264 IC50 = 8 nM T00663 C1G6KJ 137637551 IC50 = 0.6 nM T00663 CLGH04 137638967 IC50 = 3 nM T00663 CNE0Z1 137639840 IC50 = 2 nM T00663 CS3RQ4 137639936 IC50 = 4 nM T00663 CT38UG 137641182 IC50 = 24 nM T00663 CYL1R5 137643579 IC50 = 2 nM T00663 CW3IE6 137645681 IC50 = 27 nM T00663 CAY2W4 137646016 IC50 = 2 nM T00663 CGNM85 137646697 IC50 = 3 nM T00663 C5UE8A 137649558 IC50 = 175 nM T00663 CN13EH 137650943 IC50 = 0.3 nM T00663 CLN2M3 137652755 IC50 = 23 nM T00663 C8MH2Z 137654276 IC50 = 3 nM T00663 CMJF60 137655822 IC50 = 2 nM T00663 CPY1U3 137656311 IC50 = 25 nM T00663 CBI64H 137657498 IC50 = 30 nM T00663 CZFJ89 137660093 IC50 = 253 nM T00663 CA3XC2 137660956 IC50 = 200 nM T00663 CS32IR 137661932 IC50 = 10 nM T00663 CZ9BN4 138320062 IC50 = 0.107 nM T00663 C6VB3O 145925651 IC50 >= 5000 nM T00663 C2MD1Q 155513187 IC50 > 10000 nM T00663 CFV10S 155529132 IC50 = 90 nM T00663 C2CG1A 155537016 IC50 > 10000 nM T00663 D00HVA 11624601 Ki = 52 nM T00663 D02PVB 8515 IC50 = 90 nM T00663 D06PJW 25182616 IC50 = 2000 nM T00663 D0D6MH 11617559 IC50 > 16000 nM T00663 D0E3KD 447874 IC50 = 590 nM T00663 D0H2PE 10236389 IC50 = 48 nM T00663 D0J3LR 11634725 Ki = 1400 nM T00663 D0L0HG 766949 IC50 = 199.53 nM T00663 D0OZ2S 11785878 IC50 = 7300 nM T00663 D0Q3NG 11715520 Ki = 520 nM T00663 D0R3MO 46864283 IC50 > 20000 nM T00663 D0S7IE 11658882 Ki = 3300 nM T00663 D0VJ2S 57340686 IC50 = 338 nM T31186 CBHX59 5494430 IC50 > 400000 nM T31186 CGZJ49 6911989 IC50 = 43500 nM T31186 CF2Z8H 73345264 IC50 = 85000 nM T31186 C6PHF8 73345266 IC50 = 4000 nM T31186 CY07SN 73348296 IC50 = 70000 nM T31186 COC3D9 87278522 IC50 = 27000 nM T31186 CBF2I4 87278547 IC50 = 15500 nM T31186 CPHV38 87278548 IC50 = 34000 nM T31186 CK10ZE 87278578 IC50 = 45000 nM T31186 CD9M2Z 87278583 IC50 = 43500 nM T31186 CP02TE 88568566 IC50 = 25000 nM T31186 C40SKD 88568567 IC50 = 32000 nM T31186 C2SPB4 88568595 IC50 = 21500 nM T31186 C4PFH0 88568626 IC50 = 18500 nM T31186 CWUR45 88568650 IC50 = 14000 nM T31186 CVP2B8 88568651 IC50 = 28000 nM T31186 CMI83B 88568652 IC50 = 11500 nM T31186 C51NPU 90644210 IC50 = 10500 nM T31186 C8WJT2 90644211 IC50 = 10500 nM T31186 C6D0LB 90644212 IC50 = 15500 nM T31186 C76GAJ 90644213 IC50 = 30000 nM T31186 CPZ41A 90644214 IC50 = 30500 nM T31186 C9QD4R 90644215 IC50 = 32500 nM T31186 CTXP81 90644216 IC50 = 49000 nM T31186 CP3FR5 90644217 IC50 = 49000 nM T31186 CXE82I 90644218 IC50 = 16500 nM T31186 CJXI38 90644219 IC50 = 51500 nM T31186 C2VZ6T 90644220 IC50 = 55500 nM T31186 C68DLC 90644221 IC50 = 39000 nM T31186 C90QLM 90644222 IC50 = 40500 nM T31186 CMG67U 90644223 IC50 = 48500 nM T31186 C9NB5J 118719257 IC50 > 400000 nM T31186 CTZ6U9 135450598 Ki = 28 nM T31186 C9Y0KB 135501934 IC50 > 400000 nM T31186 C8DGU1 135566702 IC50 = 95 nM T31186 C48ETA 135874011 IC50 = 41 nM T31186 COAK56 135924252 IC50 = 59 nM T31186 CAN6D4 135924253 IC50 = 6580 nM T31186 CFO84Y 136086421 IC50 > 400000 nM T31186 CM8GR9 136138688 IC50 = 15500 nM T31186 CUM1R3 136138689 IC50 = 56800 nM T31186 CG4L1M 136138690 IC50 = 54500 nM T31186 CCOP90 136138691 IC50 = 10000 nM T31186 C4XN9U 136138692 IC50 = 49300 nM T31186 C5YLP4 136138694 IC50 = 5350 nM T31186 CJ73VB 136138696 IC50 = 43000 nM T31186 CGPX35 136138698 IC50 = 1590 nM T31186 CWB34M 136138700 IC50 = 125 nM T31186 CV0EY9 136138703 IC50 = 2570 nM T31186 CG3WL4 136138705 IC50 = 56 nM T31186 C9Z2WY 136138707 IC50 = 85400 nM T31186 CNL69S 136138709 IC50 = 117 nM T31186 CF5B3P 136138716 IC50 = 3600 nM T31186 CBP2Y7 136138717 IC50 = 51 nM T31186 CMN04A 136138724 IC50 = 300000 nM T31186 C2VM5F 136138725 IC50 = 1350 nM T31186 CJ9M4A 136138730 IC50 = 160 nM T31186 C7X9VW 136138737 IC50 = 16 nM T31186 CEOA02 136138748 IC50 = 3140 nM T31186 CG17QK 136168052 IC50 = 14000 nM T31186 C0G8TQ 136219232 IC50 > 400000 nM T31186 CL36PF 136239280 IC50 > 400000 nM T31186 CRD1X8 136239419 IC50 > 400000 nM T31186 CEQ20H 136244199 IC50 > 400000 nM T31186 CJQ7O0 136244535 IC50 = 400000 nM T31186 C6W2FB 136244622 IC50 = 400000 nM T31186 CI5P4A 137007090 IC50 = 200000 nM T31186 CUY95S 137007091 IC50 = 130000 nM T31186 CRBD48 137169130 IC50 = 45000 nM T31186 CP5Z9C 137169131 IC50 = 55000 nM T31186 CK7R3T 137169132 IC50 > 400000 nM T31186 C19BNM 137169134 IC50 > 400000 nM T31186 CQ67ME 137169136 IC50 > 400000 nM T31186 CIK56Z 137169159 IC50 = 5000 nM T31186 C5NAP7 137169160 IC50 = 220000 nM T31186 CLT5O9 137169161 IC50 > 400000 nM T31186 C7DQC8 137169162 IC50 > 400000 nM T31186 COB83M 137169163 IC50 = 50000 nM T31186 C9HFC1 137169164 IC50 = 100000 nM T31186 C7S6FE 137169165 IC50 = 220000 nM T31186 C7D5EQ 137169166 IC50 > 400000 nM T31186 CMAZ31 137169167 IC50 = 180000 nM T31186 C8ID1Y 145975543 Ki = 382000 nM T38996 D01XBA 5035 IC50 = 4300 nM T38996 D03JRG 46937439 IC50 = 1500 nM T38996 D0CI4A 25105704 IC50 = 21 nM T38996 D0OX9E 50902705 IC50 = 200 nM T38996 CQ0IC4 63062 IC50 = 4800 nM T38996 CW21VY 16739265 IC50 = 1 nM T38996 C17GSK 21428808 IC50 = 14000 nM T38996 C3IHB0 21428850 IC50 = 6.3 nM T38996 C9QY5H 21428857 IC50 = 22 nM T38996 CVC98H 21428895 IC50 = 4 nM T38996 C23HQA 21428932 IC50 = 5590 nM T38996 C40CFO 21428968 IC50 = 10000 nM T38996 CK90LC 21428971 IC50 = 1000 nM T38996 C8IXU1 21429000 IC50 = 10 nM T38996 CT0C3Z 25105692 IC50 = 14 nM T38996 CA7XR1 25105696 IC50 = 6000 nM T38996 C0MHU9 25105697 IC50 = 3200 nM T38996 CRG7X8 25105698 IC50 = 17 nM T38996 C54TAV 25105699 IC50 = 19 nM T38996 CIPH75 25105700 IC50 = 85 nM T38996 C9H5WS 25105701 IC50 = 32 nM T38996 CMJ14L 25105702 IC50 = 79 nM T38996 C7EW5O 25105703 IC50 = 51 nM T38996 C9J7ZI 25105705 IC50 = 20 nM T38996 CMW3Y1 25105706 IC50 = 35 nM T38996 C5MZX7 25105707 IC50 = 300 nM T38996 C2ZF1U 25105708 IC50 = 380 nM T38996 C68JBL 25105709 IC50 = 37 nM T38996 CF6P7E 25105710 IC50 = 8.9 nM T38996 C30IGQ 25105711 IC50 = 48 nM T38996 C19VQY 25105712 IC50 = 870 nM T38996 C9TX2Y 25105713 IC50 = 11 nM T38996 C48BVE 25105714 IC50 > 20000 nM T38996 C3WPU2 25105715 IC50 = 1000 nM T38996 C8XHA1 25105716 IC50 = 3400 nM T38996 CH2A5B 44138051 IC50 = 25 nM T38996 CO0V5A 44438309 IC50 = 8 nM T38996 CXB2R1 44573118 IC50 = 6.4 nM T38996 CT6FP3 44573119 IC50 = 8 nM T38996 COD46G 44573120 IC50 = 3 nM T38996 C65LXN 44573121 IC50 = 3.5 nM T38996 CD6G3I 44573130 IC50 = 4 nM T38996 C40TOA 44573131 IC50 = 3.7 nM T38996 CRC8G1 44573132 IC50 = 2 nM T38996 C8N3CM 44573176 IC50 = 5.5 nM T38996 C0D4GS 44573191 IC50 = 12 nM T38996 CSZ0W7 44573597 IC50 = 40 nM T38996 CFQA45 44573598 IC50 = 70 nM T38996 C8Q5RD 44573599 IC50 = 110 nM T38996 CC09AZ 44573641 IC50 = 120 nM T38996 C39HWT 44573687 IC50 = 4 nM T38996 CT18AS 44573688 IC50 = 18 nM T38996 CWI75L 44573689 IC50 = 12 nM T38996 C14ZEX 44573690 IC50 = 3 nM T38996 C8A4LR 44573727 IC50 = 7 nM T38996 CBM42C 44573728 IC50 = 4 nM T38996 CBCX36 44573767 IC50 = 43 nM T38996 C5BDG2 44573768 IC50 = 130 nM T38996 CQ9X2N 44573769 IC50 = 38 nM T38996 CQ62KR 44573770 IC50 = 66 nM T38996 CB2G5X 44573806 IC50 = 100 nM T38996 C1GM3U 44573807 IC50 = 11 nM T38996 CZO1C6 44573808 IC50 = 7.4 nM T38996 CEX9F5 44573809 IC50 = 10 nM T38996 CP63HT 44591888 IC50 > 20000 nM T38996 CK8GV2 44591889 IC50 = 1900 nM T38996 CHVO21 44591890 IC50 = 2100 nM T38996 CP5VO4 44591891 IC50 = 2600 nM T38996 C09BTI 44591892 IC50 = 150 nM T38996 C9E5ZV 44591930 IC50 = 150 nM T38996 CCX35M 44591931 IC50 = 4250 nM T38996 CDY58B 44591932 IC50 = 5900 nM T38996 CBHW79 44591933 IC50 > 20000 nM T38996 CFOX18 44591934 IC50 = 3400 nM T38996 C0J3UF 46938432 IC50 = 210 nM T38996 C8LAD0 46938434 IC50 = 250 nM T38996 CMB63C 46938535 IC50 = 390 nM T38996 C3GPY4 46938537 IC50 = 290 nM T38996 CNSZ76 46938539 IC50 = 335 nM T38996 CRN3Z8 46938541 IC50 = 2660 nM T38996 CYO78K 46938928 IC50 = 10 nM T38996 CB06NU 46939226 IC50 = 2500 nM T38996 CP04XW 46939227 IC50 = 11800 nM T38996 C4B2SF 46939228 IC50 = 1200 nM T38996 CV8DS2 46939229 IC50 = 870 nM T38996 CX3QE6 46939321 IC50 = 3470 nM T38996 C2K4TB 46939322 IC50 = 2800 nM T38996 CR7L9X 46939323 IC50 = 2060 nM T38996 CQI17K 46939324 IC50 = 5780 nM T38996 CJ7VN8 46939407 IC50 = 1700 nM T38996 C2ZW8V 46939408 IC50 = 2000 nM T38996 CO5X0P 46939409 IC50 = 2270 nM T38996 CY05QU 46939410 IC50 = 3500 nM T38996 C1PZM4 46939489 IC50 = 5900 nM T38996 CX49SE 46939490 IC50 = 2700 nM T38996 C14XNH 49850293 IC50 = 16 nM T38996 CF31UA 50902617 IC50 = 1700 nM T38996 C58APV 50902621 IC50 = 320 nM T38996 CPUG80 50902623 IC50 = 5500 nM T38996 C3RNG4 50902707 IC50 = 6400 nM T38996 CH38VC 50902709 IC50 > 20000 nM T38996 CRC6V8 50902786 IC50 = 12000 nM T38996 C16FQK 50902788 IC50 = 320 nM T38996 CKE14R 50902876 IC50 = 1350 nM T38996 CAJ3L1 50902978 IC50 = 1 nM T38996 C47VGW 53393916 IC50 = 20000 nM T38996 C26TVP 56593045 IC50 = 86 nM T38996 CB27OD 56593054 IC50 = 6 nM T38996 C2XP8D 56593056 IC50 = 1540 nM T38996 C3ZYA2 56593082 IC50 = 20 nM T38996 C7ENU3 56846622 IC50 = 1400 nM T38996 C1CBU4 56846623 IC50 = 760 nM T38996 CEZA46 56846640 IC50 = 75 nM T38996 C47LNP 68182778 IC50 = 250 nM T38996 CBME89 68182839 IC50 = 820 nM T38996 C6AHP7 68183060 IC50 = 16 nM T38996 COXN56 68188986 IC50 = 25 nM T38996 CUBM27 71716675 IC50 = 2 nM T38996 CWB3V1 71718136 IC50 = 6 nM T38996 CRG3Z8 73099418 IC50 > 30000 nM T38996 CV9UO7 118722101 IC50 = 315 nM T38996 C1ZJ5C 118722102 IC50 = 290 nM T38996 C9OSG5 118722103 IC50 = 120 nM T38996 CUSE27 118722104 IC50 = 18 nM T38996 C84TOB 118722105 IC50 = 6 nM T38996 CYM54A 118722106 IC50 = 17 nM T38996 C8CDM2 118722107 IC50 = 636 nM T38996 CCEL04 118722108 IC50 = 115 nM T38996 CI5MY4 118722109 IC50 = 21 nM T38996 CPF97C 118722110 IC50 = 244 nM T38996 C09UXY 118722111 IC50 = 870 nM T38996 CD73JQ 118722112 IC50 = 468 nM T38996 COU89E 118722113 IC50 = 230 nM T38996 CRB6F1 118722114 IC50 = 72 nM T38996 CMRF75 118722115 IC50 = 820 nM T38996 CBF47Z 118722116 IC50 = 115 nM T38996 C92QNG 155537801 IC50 = 21 nM T38996 CVU9P7 155540036 IC50 = 1200 nM T38996 D07JMN 94459 IC50 = 3600 nM T38996 D07RPV 65490 IC50 = 21 nM T38996 D0IV2E 5280592 IC50 > 1000 nM T38996 D0T3HK 70517 IC50 = 3600 nM T43920 D0C2II 4100 IC50 = 20 nM T43920 D0E1SW 1986 Ki = 0.8 nM T43920 CG2Q9U 66824 Ki = 0.3 nM T43920 CJR96B 72879 IC50 = 1000000 nM T43920 C04JEX 73702 IC50 = 1000000 nM T43920 CCK5Y6 133125 IC50 = 550 nM T43920 C8KN4F 133683 IC50 = 20 nM T43920 C2GA7W 195627 IC50 = 730 nM T43920 CZL4G0 232992 Ki = 584 nM T43920 CPA95I 232993 Ki = 146 nM T43920 CD23RS 641380 IC50 = 550 nM T43920 CM5FP2 3769607 IC50 = 20 nM T43920 C83URK 4343109 IC50 = 20 nM T43920 CH62SB 5325614 IC50 = 480 nM T43920 C18GCW 13754314 Ki = 258 nM T43920 C4JD1S 13755238 Ki = 44 nM T43920 CA8D6Y 13755239 Ki = 107 nM T43920 CX4V9O 13904667 IC50 = 20 nM T43920 C28TEH 13904668 IC50 = 18 nM T43920 C7Q1BO 13904669 IC50 = 14 nM T43920 CE51MD 13904671 IC50 = 50 nM T43920 CXK68I 13904672 IC50 = 50 nM T43920 C7YX0N 15665951 IC50 = 370 nM T43920 C6DU3A 15665952 IC50 = 390 nM T43920 CK8BI3 15665953 IC50 = 520 nM T43920 C0ASB7 15665954 IC50 = 910 nM T43920 CL35KY 15665955 IC50 = 440 nM T43920 CW6LI5 15665958 IC50 = 450 nM T43920 CK72NU 15665961 IC50 = 310 nM T43920 CVSL38 15665962 IC50 = 940 nM T43920 CRXL21 15665963 IC50 = 230 nM T43920 C89TJU 15665964 IC50 = 910 nM T43920 C3NZO2 15665965 IC50 = 520 nM T43920 C2QL3W 15665966 IC50 = 520 nM T43920 CN7J6P 44343745 IC50 = 84 nM T43920 C6KUJ0 44343753 IC50 = 770 nM T43920 C5EIQ0 59552403 Ki = 0.2 nM T43920 CQN51D 118724498 IC50 = 441720 nM T43920 C8F9DB 135898802 IC50 = 37 nM T43920 CR17HF 155510806 Ki = 0.2 nM T43920 C2H9WX 155554455 Ki = 0.2 nM T43920 D06LVE 22784 Ki = 0.2 nM T43920 D09QHC 7370 IC50 = 2000 nM T97587 CTA32V 9831270 IC50 = 49 nM T97587 C7J3ZW 9847562 IC50 = 1.4 nM T97587 CV9X1Q 9871831 IC50 = 3.7 nM T97587 CSY94G 9893920 IC50 = 0.87 nM T97587 C5BXR9 9960341 IC50 = 1.6 nM T97587 C8J2IQ 9961835 IC50 = 0.2 nM T97587 C8AJ2G 9985610 IC50 = 0.64 nM T97587 C3VX4B 10175373 IC50 = 99 nM T97587 C1BK6W 10348108 IC50 = 20 nM T97587 CS12LU 10369544 IC50 = 0.5 nM T97587 C4D8CL 10415520 IC50 = 0.7 nM T97587 C4TGS8 15984101 IC50 = 0.51 nM T97587 CNG3Y6 20828691 IC50 = 0.07 nM T97587 C5XI2B 23647822 IC50 = 9.2 nM T97587 CV87US 23647823 IC50 = 106 nM T97587 C4NZC8 23647824 IC50 = 769 nM T97587 C7K6VJ 23647825 IC50 = 49 nM T97587 CTV02H 23647826 IC50 = 282 nM T97587 CD36OZ 23647827 IC50 = 216 nM T97587 CB54AV 23647828 IC50 = 15 nM T97587 CIN2D4 23647829 IC50 = 8.4 nM T97587 CDC59X 23647830 IC50 = 13 nM T97587 C23IKQ 23647831 IC50 = 1.3 nM T97587 CT19JC 23647832 IC50 = 1.3 nM T97587 C7RB6T 23647833 IC50 = 9.8 nM T97587 CUYM23 23647834 IC50 = 1.7 nM T97587 C0HD6M 23647835 IC50 = 95 nM T97587 CUP79Y 24875357 IC50 = 237 nM T97587 CG17MD 25147778 IC50 = 1.6 nM T97587 CS98GW 25242385 IC50 = 2.8 nM T97587 C78USC 44157321 IC50 = 0.09 nM T97587 C86VTZ 44157395 IC50 = 0.1 nM T97587 CF01CW 44157473 IC50 = 0.1 nM T97587 C5QDR9 44157717 IC50 = 0.2 nM T97587 CJ1GX4 44157718 IC50 = 0.3 nM T97587 CPI0L1 44270826 IC50 = 550 nM T97587 C2ITA9 44270830 IC50 = 330 nM T97587 CAYN82 44270836 IC50 = 160 nM T97587 CTU6S9 44270842 IC50 = 44 nM T97587 C9ONK1 44271028 IC50 = 35 nM T97587 CXM20K 44271069 IC50 = 0.1 nM T97587 CMX53A 44271083 IC50 = 2.7 nM T97587 CAU67L 44271148 IC50 = 3.9 nM T97587 CU2DL4 44271164 IC50 = 1.8 nM T97587 CR94DM 44271244 IC50 = 19 nM T97587 CR06WP 44271256 IC50 = 112 nM T97587 CKP31U 44271273 IC50 = 5 nM T97587 C0W9BH 44446215 IC50 = 123 nM T97587 CE29ZY 44446216 IC50 = 135 nM T97587 CT9G8Q 44446217 IC50 = 170 nM T97587 CS36EO 44446218 IC50 = 152 nM T97587 C02NZQ 44446219 IC50 = 353 nM T97587 C2S7QF 44446220 IC50 = 327 nM T97587 CV4L9G 44446221 IC50 = 450 nM T97587 CQXG81 44446222 IC50 = 143 nM T97587 CC8HU7 44446223 IC50 = 239 nM T97587 CV49GF 44446224 IC50 = 75 nM T97587 CP0TH8 44446225 IC50 = 179 nM T97587 CDM45Z 44446226 IC50 = 235 nM T97587 C1WRY6 44446227 IC50 = 222 nM T97587 CX6T3Z 44446228 IC50 = 130 nM T97587 CL9DG6 44446229 IC50 = 76 nM T97587 CWTX92 44446230 IC50 = 69 nM T97587 CD0QV3 44446231 IC50 = 67 nM T97587 COXP59 44446232 IC50 = 101 nM T97587 C8T6CM 44446233 IC50 = 19 nM T97587 C08SHV 44446234 IC50 = 67 nM T97587 C56TUJ 44446236 IC50 = 124 nM T97587 C1G6AZ 44446238 IC50 = 80 nM T97587 C7USF6 44446240 IC50 = 200 nM T97587 C7IU9H 44446241 IC50 = 196 nM T97587 C7R4QZ 44446243 IC50 = 28 nM T97587 C79HBR 44446248 IC50 = 1122 nM T97587 CG83CS 44446251 IC50 = 6807 nM T97587 C9UZ0X 44446256 IC50 = 4318 nM T97587 CF5DT9 44446259 IC50 = 510 nM T97587 C5ZQ3C 44446261 IC50 = 42 nM T97587 C9IS1C 44455093 IC50 = 285 nM T97587 CB51GK 44455095 IC50 = 2535 nM T97587 CX23CH 44455169 IC50 = 2100 nM T97587 CB9T2Z 44571247 IC50 = 831 nM T97587 C1R5VH 44571248 IC50 = 198 nM T97587 CBK28E 44571249 IC50 = 164 nM T97587 COG41E 44571293 IC50 = 50 nM T97587 CS80NQ 44571294 IC50 = 19 nM T97587 CP6M5Y 44571295 IC50 = 19 nM T97587 CB26YW 44587963 IC50 = 7.5 nM T97587 CVTM09 44587964 IC50 = 4.8 nM T97587 CG2RX4 44587965 IC50 = 12 nM T97587 C52MPU 44588004 IC50 = 2.8 nM T97587 C05GKL 44588445 IC50 = 2.9 nM T97587 CT81MC 44588480 IC50 = 2.2 nM T97587 C3KSC4 44588481 IC50 = 44 nM T97587 C0JS4X 44588482 IC50 = 1.9 nM T97587 CDPT75 44588524 IC50 = 630 nM T97587 CUCZ38 44588525 IC50 = 3.5 nM T97587 C05LYK 44588526 IC50 = 688 nM T97587 CT8PH7 45485800 IC50 = 0.34 nM T97587 CHP37W 45485803 IC50 = 0.16 nM T97587 CLFJ36 45485807 IC50 = 0.11 nM T97587 CTR5Z7 46229904 IC50 = 0.22 nM T97587 C3XAQ6 46229905 IC50 = 0.81 nM T97587 CSP19C 46229906 IC50 = 0.55 nM T97587 C40XVP 46229907 IC50 = 0.08 nM T97587 CI2O9L 46229908 IC50 = 0.25 nM T97587 C7F0MK 46229909 IC50 = 0.35 nM T97587 CO4D9I 46229910 IC50 = 0.08 nM T97587 CVL02P 46229911 IC50 = 0.42 nM T97587 CG7V9S 46229912 IC50 = 0.25 nM T97587 C0ML2V 46229913 IC50 = 0.13 nM T97587 C42KWF 46229914 IC50 = 0.13 nM T97587 CTK82C 46229915 IC50 = 0.11 nM T97587 CM43CI 46229916 IC50 = 0.13 nM T97587 CE4Q9R 46229917 IC50 = 0.16 nM T97587 C93TOU 46229918 IC50 = 0.14 nM T97587 CJX9A5 46229919 IC50 = 0.16 nM T97587 C93JUZ 49865755 IC50 = 2700 nM T97587 CQEB67 49865756 IC50 = 8300 nM T97587 CAO82G 49865757 IC50 = 9500 nM T97587 C5CPE8 49865758 IC50 = 6300 nM T97587 CZ4SH8 49865759 IC50 = 100 nM T97587 CYG30P 49865760 IC50 = 9000 nM T97587 CT5DJ6 49865761 IC50 = 6300 nM T97587 CX8C0E 49865762 IC50 = 7900 nM T97587 CI4Q6S 49865763 IC50 = 8700 nM T97587 CVP7M6 49865764 IC50 = 500 nM T97587 COSD80 49865765 IC50 = 1400 nM T97587 CB2RH6 49865766 IC50 = 1200 nM T97587 C7QNM0 49865842 IC50 = 2100 nM T97587 CT8H9I 49865843 IC50 = 1500 nM T97587 CL0O3V 49865844 IC50 = 1100 nM T97587 CMVB16 49865845 IC50 = 4400 nM T97587 CV3XC8 49865895 IC50 = 1500 nM T97587 CHI31D 49865896 IC50 = 6600 nM T97587 C5MK9C 49865897 IC50 = 1200 nM T97587 C4CR0M 49865898 IC50 = 300 nM T97587 CE2H9O 49865899 IC50 = 600 nM T97587 C1MJI2 49865946 IC50 = 700 nM T97587 C7QIX2 49865947 IC50 = 600 nM T97587 CZE86G 49865948 IC50 = 3000 nM T97587 C7TUL0 49865949 IC50 = 600 nM T97587 CP74MO 49865950 IC50 = 700 nM T97587 C8D7SR 49865996 IC50 = 2800 nM T97587 C6ZFN2 49865997 IC50 = 600 nM T97587 C3HNC7 49865998 IC50 = 1500 nM T97587 CPO1L3 49865999 IC50 = 900 nM T97587 CEK6Z9 49866051 IC50 = 200 nM T97587 C0G5SY 49866052 IC50 = 1500 nM T97587 CUW64X 49866053 IC50 = 500 nM T97587 C41GCZ 49866107 IC50 = 700 nM T97587 C4C7EB 49866108 IC50 = 400 nM T97587 C1NB5E 49866109 IC50 = 1000 nM T97587 C87SXF 49866110 IC50 = 2600 nM T97587 CK5ZC9 49866111 IC50 = 3400 nM T26463 D02ILH 341 Ki = 830 nM T26463 D05RQB 457964 EC50 = 2000 nM T26463 CZP5J2 3415 IC50 > 20000 nM T26463 C4DTF0 6665 IC50 > 500000 nM T26463 CLO15X 67277 IC50 = 32000 nM T26463 CQ87XE 72187 IC50 = 13400 nM T26463 CMR72P 127307 Ki = 14400 nM T26463 CQ1XM2 149664 Ki = 1400 nM T26463 C7Y0CH 238747 IC50 = 28000 nM T26463 C6NE8Z 389513 Ki = 1000 nM T26463 CO6A2E 451388 IC50 = 1000 nM T26463 C9L0ZN 481497 IC50 > 100000 nM T26463 CF2YG0 481498 IC50 = 63000 nM T26463 C9I6LT 481500 IC50 = 18000 nM T26463 CY24WL 481501 IC50 > 100000 nM T26463 C9U7BA 481504 IC50 = 93000 nM T26463 CU3P0Y 484047 IC50 > 40000 nM T26463 CL4X0H 491953 IC50 > 50000 nM T26463 CP8ZJ7 491954 IC50 = 26000 nM T26463 C61SXL 492406 IC50 > 40000 nM T26463 CXD5F2 496192 IC50 = 85000 nM T26463 CM6J2G 496196 Ki = 5000 nM T26463 CDW6L4 497307 IC50 = 480 nM T26463 CZJP19 497308 IC50 > 100000 nM T26463 CX9ZP0 497310 IC50 = 800 nM T26463 C74SZP 497311 IC50 = 15 nM T26463 CZ1A8T 503580 IC50 > 40000 nM T26463 C8UMS5 3005246 Ki = 36000 nM T26463 C3E1ZI 3012981 IC50 > 100000 nM T26463 C1FXQ4 5466207 Ki = 2600 nM T26463 C8F1DN 6482394 IC50 > 40000 nM T26463 C6OF2J 6914644 IC50 > 100000 nM T26463 CQP57I 9802791 IC50 > 500000 nM T26463 CF5TC2 9805202 IC50 = 5000 nM T26463 CHT36N 9828287 IC50 = 3000 nM T26463 C47XQV 9938296 IC50 = 5000 nM T26463 CA9Q4Z 10078740 IC50 = 1900 nM T26463 C1JN2O 10120254 IC50 > 10000 nM T26463 C7SO4T 10144617 IC50 > 10000 nM T26463 C3B2KX 10185481 IC50 > 10000 nM T26463 CB5O0Q 10185854 IC50 > 50000 nM T26463 CDQ6H2 10209030 IC50 > 10000 nM T26463 C58FZS 10230222 IC50 > 10000 nM T26463 C5AXK6 10230544 IC50 > 10000 nM T26463 CZ48MN 10385259 IC50 = 66000 nM T26463 C5O4HY 10647065 Ki = 7840 nM T26463 CNKU56 10893485 IC50 > 50000 nM T26463 CG2KN4 10918740 Ki = 156000 nM T26463 CB98DN 11014401 IC50 = 4300 nM T26463 CIYW64 11686018 IC50 > 10000 nM T26463 C7Z5LI 11764703 Ki = 548000 nM T26463 CUB20Q 15949381 IC50 > 10000 nM T26463 CEL84W 15956783 IC50 > 10000 nM T26463 COP0D7 15956784 IC50 > 10000 nM T26463 C51OVS 15956785 IC50 > 10000 nM T26463 CIU52S 21589997 IC50 > 12500 nM T26463 C0L2TF 23725128 IC50 > 100000 nM T26463 C1P2KY 24771829 EC50 = 350000 nM T26463 CO25RL 25000921 IC50 > 100000 nM T26463 CG9S8U 44396484 IC50 = 8000 nM T26463 CSQ5K2 44396511 Ki = 3750 nM T26463 CC2AE1 44396529 IC50 > 500000 nM T26463 C0GDR1 44396563 IC50 > 500000 nM T26463 CK8ZW1 44396581 IC50 > 500000 nM T26463 CE04QD 44396595 IC50 > 500000 nM T26463 CZ6DX1 44412144 IC50 = 1900 nM T26463 CGM62X 44412145 IC50 = 3300 nM T26463 CZ18LU 44412189 IC50 = 8900 nM T26463 C3MSG6 44412212 IC50 = 7900 nM T26463 C3JG6P 44412241 IC50 = 2300 nM T26463 C2U6NS 44412250 IC50 = 3500 nM T26463 C1WGS5 44412370 IC50 = 25000 nM T26463 CX1GZ9 44412378 IC50 = 19900 nM T26463 C1XN2M 44412379 IC50 = 19700 nM T26463 C7ZKR6 44412431 IC50 = 6900 nM T26463 CD72OK 44412489 IC50 = 21000 nM T26463 C5V2QB 44412490 IC50 = 3700 nM T26463 C6V1JG 44604808 IC50 > 20000 nM T26463 CQ1N2M 44605023 IC50 > 20000 nM T26463 CNK9D2 44607341 IC50 > 20000 nM T26463 CCQS46 46830304 IC50 > 20000 nM T26463 CVAT67 53317946 IC50 > 500000 nM T26463 CT7D5O 53320320 IC50 > 100000 nM T26463 CK6RI2 53324652 IC50 > 100000 nM T26463 CY32HG 54677477 IC50 > 10000 nM T26463 C0ZG2V 54709839 IC50 > 200000 nM T26463 CLT3Q8 54716246 IC50 > 10000 nM T26463 CU9M3O 56832906 IC50 > 200000 nM T26463 CDS0C6 66825540 IC50 > 500000 nM T26463 CH1S3G 71548918 IC50 > 25000 nM T26463 CFG02R 73669532 IC50 > 500000 nM T26463 C9DY6C 76318645 IC50 = 45000 nM T26463 CQ29OX 76325888 IC50 > 500000 nM T26463 CSJ2W1 86302310 EC50 = 80000 nM T26463 C6ZY2A 90654414 EC50 > 500000 nM T26463 CXN6B4 90654415 EC50 > 500000 nM T26463 CSH13R 90654416 EC50 > 500000 nM T26463 C0PC8E 90654417 EC50 = 250000 nM T26463 CR2OE7 90654418 EC50 > 500000 nM T26463 CRP0L2 90654419 EC50 = 70000 nM T26463 C1Y5EA 90654420 EC50 = 410000 nM T26463 CW1B9O 90654421 EC50 > 500000 nM T26463 CU4G2C 117940941 IC50 = 20200 nM T26463 CT6M7E 135435051 IC50 = 46000 nM T26463 CW0CR6 135435052 Ki = 44000 nM T26463 CD38IL 135435084 Ki = 7500 nM T26463 CD5QA6 135435086 Ki = 1760000 nM T26463 C63ONQ 135435181 IC50 > 50000 nM T26463 CZ4GP6 135446244 IC50 > 10000 nM T26463 CUBV31 135485600 IC50 = 2500 nM T26463 CZH2Y8 135537671 Ki = 2300 nM T26463 C1EDK4 136030640 IC50 > 100000 nM T26463 C2H5PQ 136215370 Ki = 1 nM T26463 C8BJ0A 134007 EC50 = 4000 nM T26463 C0UQH8 516384 EC50 = 8000 nM T26463 C91IWY 516389 EC50 = 3000 nM T26463 CID8Z7 516390 EC50 = 5000 nM T26463 CLU03S 516391 EC50 = 3000 nM T26463 C5P8LV 516396 EC50 = 4000 nM T26463 CT01UL 516397 EC50 = 1000 nM T26463 CP5BZ4 5271338 EC50 = 7000 nM T26463 D02DLW 5997 IC50 > 500000 nM T99089 D05ROI 44462760 IC50 = 0.4 nM T99089 D07POC 176870 IC50 = 60 nM T99089 D09GDD 11167602 IC50 = 1.5 nM T99089 D09XZB 123631 IC50 = 2000 nM T99089 D0AZ3C 5291 IC50 > 100000 nM T99089 D0J9ZR 4477 IC50 > 100000 nM T99089 D0K8KX 5280343 IC50 = 7589 nM T99089 D0TK7R 50922675 IC50 = 0.3 nM T99089 D0W5HK 216239 IC50 = 1 nM T99089 D0Y9EW 42611257 IC50 = 4 nM T99089 D02UFQ 11620908 IC50 > 10000 nM T99089 D03AND 11656518 IC50 = 20 nM T99089 D03LWG 53235510 IC50 = 4142 nM T99089 D04AHQ 71721540 IC50 = 1.5 nM T99089 D04MXN 56846693 IC50 = 82 nM T99089 D0E3TC 44259 IC50 = 4.5 nM T99089 D0F5JZ 24180719 Ki = 2.6 nM T99089 D0K0YC 9826528 IC50 = 6 nM T99089 D0M5XN 89670174 IC50 = 23 nM T99089 D0O2FN 16222096 IC50 = 1.8 nM T99089 D0T4QA 90456533 IC50 = 0.4 nM T99089 D0Z2FD 56931136 IC50 = 6 nM T99089 D04SWX 56924694 IC50 = 270 nM T99089 D0B7VP 46198319 IC50 = 26 nM T99089 D0T3ME 156422 IC50 = 83.4 nM T99089 CB37VR 5034 IC50 = 29.6 nM T99089 C63WLY 89644 IC50 > 10 ug.mL-1 T99089 C5JE2Z 104860 IC50 = 6.7 ug.mL-1 T99089 CI1NA5 159926 IC50 = 6.4 ug.mL-1 T99089 CYBA43 177458 IC50 > 10 ug.mL-1 T99089 C9VW8M 449054 IC50 > 16000 nM T99089 COI61Y 660701 IC50 > 100000 nM T99089 CG1YH4 690397 IC50 = 830 nM T99089 C41EFM 691845 IC50 = 670 nM T99089 C9IL3X 697391 IC50 = 6100 nM T99089 CKX97G 698872 IC50 = 730 nM T99089 CRB31Z 741849 IC50 = 2100 nM T99089 CH9O0J 751729 IC50 > 100000 nM T99089 C82CGY 777751 IC50 > 100000 nM T99089 C4D2FR 817983 IC50 = 30110 nM T99089 C2SW3J 838432 IC50 = 740 nM T99089 C62VFD 903392 IC50 = 2010 nM T99089 C3ZTU4 985658 IC50 = 11080 nM T99089 CP9L1G 1006450 IC50 = 2230 nM T99089 CRP32Q 1006453 IC50 = 3450 nM T99089 CJF53S 1016049 IC50 = 1020 nM T99089 CF80DN 1032682 IC50 > 100000 nM T99089 CD12EO 1040090 IC50 > 100000 nM T99089 C26TIY 1088625 IC50 > 100000 nM T99089 CGP84Q 1102777 IC50 = 470 nM T99089 C6X1YI 1124092 IC50 = 4010 nM T99089 CMS5J7 1207521 IC50 = 1800 nM T99089 C01WYP 1220545 IC50 = 1160 nM T99089 CJ7M4N 1236338 IC50 > 100000 nM T99089 COH8I7 1496173 IC50 = 630 nM T99089 CG3F6Y 1684063 IC50 = 2160 nM T99089 CKR8H5 1684186 IC50 = 770 nM T99089 CEPI38 1737233 IC50 = 1540 nM T99089 CPI69L 1740003 IC50 = 4110 nM T99089 C17WVD 1771530 IC50 = 2490 nM T99089 CD76PH 1774314 IC50 = 4020 nM T99089 CKG4R9 1774320 IC50 = 3240 nM T99089 CU0O5C 1776533 IC50 = 4750 nM T99089 CLOW51 1776608 IC50 = 1600 nM T99089 CN6O3E 1793969 IC50 = 1650 nM T99089 CS2JL0 1814300 IC50 = 310 nM T99089 C3B5PI 1814302 IC50 = 970 nM T99089 CCI76Z 1814304 IC50 = 820 nM T99089 CN3G5B 1814306 IC50 = 440 nM T99089 CG02RT 1814308 IC50 = 1140 nM T99089 CC54MB 1814310 IC50 = 500 nM T99089 C27FVB 2133813 IC50 = 570 nM T99089 CZ6EV4 2133817 IC50 = 100 nM T99089 C5GYO1 2730801 IC50 = 320 nM T99089 CZE13I 2816786 IC50 = 400 nM T99089 CJ5UL8 2855606 IC50 > 100000 nM T99089 CMG0F6 2961623 IC50 = 400 nM T99089 CB4QI1 2966018 IC50 = 3000 nM T99089 CHC5I0 2971839 IC50 = 1800 nM T99089 CFY1D0 2974957 IC50 = 17 nM T99089 CW3DC7 2977311 IC50 = 800 nM T99089 C4RH3J 3106064 IC50 = 1720 nM T99089 C1GTF0 3143674 IC50 > 100000 nM T99089 C2HUN0 3235666 IC50 > 100000 nM T99089 C2H0KF 3718048 IC50 = 380 nM T99089 C73RZL 3937063 IC50 = 900 nM T99089 C4FDE6 4647084 IC50 > 100000 nM T99089 CDQ3M7 5359485 IC50 = 1.6 ug.mL-1 T99089 C54BYP 5360741 IC50 = 4.8 ug.mL-1 T99089 CTFA62 5521855 IC50 = 37480 nM T99089 C6J1DO 5716697 IC50 = 900 nM T99089 CE0SB4 5753911 IC50 > 50000 nM T99089 CXZ30D 5753913 IC50 = 11360 nM T99089 CFO1B9 5753916 IC50 = 4600 nM T99089 CM87HL 5753919 IC50 = 57890 nM T99089 CK08PH 5753938 IC50 = 10910 nM T99089 CFSD40 6510636 IC50 = 17360 nM T99089 C6KN7F 6877485 IC50 > 100000 nM T99089 C9U7GE 7718544 IC50 = 340 nM T99089 CSX8V7 7897116 IC50 = 400 nM T99089 C5GE7T 9917045 IC50 = 7200 nM T99089 C5E7HJ 10217017 IC50 = 2 nM T99089 C7S9KW 10222594 IC50 = 40 nM T99089 CXC91Z 11167118 IC50 = 280 nM T99089 CC6VK1 11236275 IC50 = 310 nM T99089 CM30TC 11387552 EC50 = 100 nM T99089 C0Z9YQ 11433057 EC50 = 100 nM T99089 CZ73AJ 11476663 IC50 = 1 nM T99089 CD6QW4 11494370 IC50 = 20000 nM T99089 CU30IV 11501142 IC50 = 10000 nM T99089 CFMS75 11501578 IC50 = 27000 nM T99089 CWZS50 11501869 IC50 = 37000 nM T99089 CB6ME8 11503895 IC50 = 47 nM T99089 C7Q5JI 11516491 IC50 = 3 nM T99089 CUDR26 11518018 IC50 = 12 nM T99089 C8AY3B 11518031 IC50 = 0.46 nM T99089 C6D9OT 11522875 IC50 = 8000 nM T99089 C3LGD4 11523321 IC50 = 3.46 nM T99089 CXP87N 11523639 IC50 = 950 nM T99089 CL7X4Q 11530963 IC50 = 40000 nM T99089 CX4D8Z 11532611 IC50 = 16 nM T99089 CCU2B0 11544514 IC50 = 45000 nM T99089 CJ23SH 11545064 IC50 = 5200 nM T99089 C6I9YN 11545261 IC50 = 0.33 nM T99089 CP3JY9 11546962 IC50 = 8300 nM T99089 C7H9FD 11551727 IC50 = 26000 nM T99089 C60ORJ 11552560 IC50 = 4500 nM T99089 CCQ4L1 11552561 IC50 = 34000 nM T99089 C0OHL1 11561411 IC50 = 1240 nM T99089 CAXP50 11566757 IC50 = 0.87 nM T99089 C4NS5D 11573300 IC50 > 100000 nM T99089 COFT94 11573823 IC50 = 65000 nM T99089 CX2B3N 11574129 IC50 = 3000 nM T99089 C34QRP 11574273 IC50 = 790 nM T99089 CPLH36 11574625 IC50 = 2300 nM T99089 C03WNJ 11574718 IC50 = 26000 nM T99089 CE30QF 11574855 IC50 = 7 nM T99089 C4O0VX 11580569 IC50 = 14000 nM T99089 C1HCK9 11581360 IC50 = 8800 nM T99089 CX4W5I 11583265 IC50 > 100000 nM T99089 CEM6P4 11583341 IC50 = 24 nM T99089 CKWN65 11588629 IC50 = 1300 nM T99089 C40YLN 11590139 IC50 = 39000 nM T99089 CK63UF 11595532 IC50 = 4000 nM T99089 C28FJS 11597486 IC50 = 61 nM T99089 CZGU14 11601866 IC50 = 1.4 nM T99089 CQ9DC4 11602668 IC50 = 33000 nM T99089 CTB45J 11603925 IC50 = 14000 nM T99089 C8YIS9 11604883 IC50 = 333 nM T99089 CZD5J8 11605467 IC50 = 497 nM T99089 C8A2LO 11610758 IC50 = 1.2 nM T99089 CP62YV 11616462 IC50 = 0.02 nM T99089 CBWP68 11624720 IC50 = 3000 nM T99089 C0OGU9 11624721 IC50 = 9800 nM T99089 CS17RF 11624965 IC50 = 0.22 nM T99089 CSM62L 11626920 IC50 = 27 nM T99089 C9K7QI 11632277 IC50 = 38000 nM T99089 CH7YA4 11633452 IC50 > 100000 nM T99089 CU98ZH 11633786 IC50 = 15 nM T99089 CS2K5N 11634109 IC50 = 192 nM T99089 C34HID 11634929 IC50 = 135 nM T99089 CMSA04 11639637 IC50 = 0.34 nM T99089 C4RX1P 11639649 IC50 = 5200 nM T99089 C6L4EZ 11645222 IC50 = 33000 nM T99089 C8Y6CU 11653652 IC50 = 0.03 nM T99089 C24KYX 11659444 IC50 = 77 nM T99089 C3PT8Y 11660026 IC50 = 74000 nM T99089 C8J7IA 11660270 IC50 = 0.39 nM T99089 C40LAT 11660528 IC50 = 3800 nM T99089 CAW41S 11667128 IC50 = 2.4 nM T99089 CT29KC 11667144 IC50 = 4000 nM T99089 CULF07 11676720 IC50 = 16 nM T99089 C4Q2OK 11681939 IC50 > 100000 nM T99089 CK42CI 11682654 IC50 = 3500 nM T99089 C8JW5Z 11696578 IC50 = 1120 nM T99089 C4WM6K 11697289 IC50 = 26 nM T99089 C6LQ9H 11702547 IC50 = 4200 nM T99089 CZ4E6K 11703339 IC50 = 12 nM T99089 C86TWZ 11704203 IC50 = 37000 nM T99089 CE30QZ 11704625 IC50 = 14 nM T99089 CQ2P3D 11704845 IC50 = 45 nM T99089 CAL4G1 11705461 IC50 = 90 nM T99089 CI0CM8 11709835 IC50 = 1400 nM T99089 CW5H0K 11710340 IC50 = 3000 nM T99089 CVR15H 11710382 IC50 = 26000 nM T99089 CGI1D9 11717001 Ki = 0.13 nM T99089 C1DF0R 11717449 IC50 = 490 nM T99089 C8O1MN 11719900 IC50 = 45 nM T99089 C5YXA3 11720025 IC50 > 100000 nM T99089 C2EX5W 11737996 IC50 = 900 nM T99089 C8MOK3 11750699 IC50 = 25 nM T99089 C39TYN 11841124 IC50 > 100000 nM T99089 CHAD78 11841127 IC50 > 100000 nM T99089 CA2LF8 11947957 IC50 = 236.7 nM T99089 CDGF78 15282555 IC50 = 2700 nM T99089 C7LB4I 15949613 IC50 = 900 nM T99089 CS3EB6 16044861 IC50 = 1.4 nM T99089 C0Z6VU 16045086 IC50 = 1 nM T99089 CA1T2U 16045087 IC50 = 16 nM T99089 C04TRQ 16045682 IC50 = 3 nM T99089 C35ILP 16045759 IC50 = 52 nM T99089 CQ4O0Y 16045761 IC50 = 3 nM T99089 C1VS7Q 16045839 IC50 = 1.1 nM T99089 CCFT24 16046014 IC50 = 1.4 nM T99089 CE43QM 16064288 IC50 = 130 nM T99089 CELY15 16064449 IC50 = 780 nM T99089 C8UOX0 16064748 IC50 = 480 nM T99089 CFKE48 16064750 IC50 = 120 nM T99089 CC7QD3 16064891 IC50 = 210 nM T99089 CLG6R7 16064892 IC50 = 42 nM T99089 C0C2QW 16064893 IC50 = 620 nM T99089 CM3A7W 16066694 IC50 = 19 nM T99089 CVE6C8 16086088 IC50 = 27 nM T99089 CU5Y7N 16101466 IC50 = 199 nM T99089 C5VPH9 16129448 IC50 > 10000 nM T99089 CZ08YH 16214904 IC50 = 53 nM T99089 CFN5D6 16223710 IC50 = 5.1 nM T99089 CB65EI 16223711 IC50 = 45 nM T99089 C8EF0N 16223900 IC50 = 49 nM T99089 C45HCU 16223901 IC50 = 93 nM T99089 CVIU65 16223902 IC50 = 1550 nM T99089 C1L8UO 16224102 IC50 = 933 nM T99089 CK5TJ0 16678105 IC50 = 17.4 nM T99089 C0EV8X 19355820 IC50 > 1000 nM T99089 C6AV4G 21023795 IC50 = 14 nM T99089 C4AK5J 21037180 IC50 = 25 nM T99089 C9YR7W 21037208 IC50 = 68 nM T99089 C8ID6R 21037243 EC50 > 10000 nM T99089 C2V1EQ 21037245 EC50 > 10000 nM T99089 CZ23BW 21037364 IC50 = 140 nM T99089 CJ4E1M 22040403 IC50 = 2700 nM T99089 C8VJ3A 22040410 IC50 = 1300 nM T99089 CHFO54 22040436 EC50 = 7000 nM T99089 CJ3UH0 22040625 IC50 = 11 nM T99089 C02DQZ 22040627 IC50 = 11 nM T99089 CCA1D7 22040647 IC50 = 39 nM T99089 C4RP8N 22040656 IC50 = 63 nM T99089 C9A4LW 22040760 IC50 = 13 nM T99089 CI3V6C 22040802 IC50 = 130 nM T99089 C9WU0J 22040805 IC50 = 2400 nM T99089 CDN61H 22040847 IC50 = 39 nM T99089 C3SX8H 22040857 IC50 = 9000 nM T99089 C6NM3T 22040925 IC50 = 140 nM T99089 CC84UT 22040937 IC50 = 1900 nM T99089 CZM5W1 22040941 IC50 = 8 nM T99089 C6FMB5 22040978 IC50 = 500 nM T99089 CRJ4H3 22041111 IC50 = 7700 nM T99089 CO37NP 22041112 IC50 = 4400 nM T99089 C4UMZ2 22041119 IC50 = 300 nM T99089 CI5KM3 22041171 IC50 = 88 nM T99089 C51FDU 22041175 IC50 = 26 nM T99089 CR3G0K 22041260 EC50 = 3200 nM T99089 C69BSO 22041261 IC50 = 28 nM T99089 CGX61W 22041319 IC50 = 45 nM T99089 CDM83W 22057968 IC50 = 2 nM T99089 CQJ59G 22185379 IC50 = 8 nM T99089 CFMT70 22185475 IC50 = 6 nM T99089 C0X7MW 22185489 IC50 = 13 nM T99089 CL5D8X 22256705 IC50 = 33 nM T99089 CXS28L 22918445 IC50 = 338 nM T99089 C7HUS0 23585267 IC50 = 32 nM T99089 CHQ23N 23585318 IC50 = 26 nM T99089 COSI68 23585320 IC50 = 20 nM T99089 CR2AN0 24180721 IC50 > 100000 nM T99089 CC6JO7 24737670 IC50 = 19 nM T99089 CZ8BQ6 24737709 IC50 = 110 nM T99089 C4GUC1 24738493 IC50 = 316 nM T99089 CLH3G9 24738495 IC50 = 718 nM T99089 CCO8T6 24738496 IC50 = 407 nM T99089 CHU49V 24757938 IC50 = 40 nM T99089 C7YG1N 24759534 IC50 = 550 nM T99089 CCPS81 24764502 IC50 > 35000 nM T99089 CC13WT 24768568 IC50 = 99 nM T99089 CCP2M3 24822704 IC50 = 32 nM T99089 CA4D9N 24829351 IC50 = 6 nM T99089 CCS58O 24863072 IC50 = 70 nM T99089 C6R4ZU 24863189 IC50 = 310 nM T99089 C6C2GX 24863500 IC50 = 110 nM T99089 CYVB83 24863584 IC50 = 18 nM T99089 CQ15ML 24863670 IC50 = 21 nM T99089 C4XZ3N 24863671 IC50 = 270 nM T99089 CU53DP 24878669 IC50 = 1400 nM T99089 C6Q4FC 24878670 IC50 = 92000 nM T99089 CUIS63 24878671 IC50 = 650 nM T99089 CGKA14 24878672 IC50 = 2500 nM T99089 C0P4HO 24879140 IC50 = 2900 nM T99089 CBUG02 24879141 IC50 = 1160 nM T99089 CSJ7T8 24879142 IC50 = 16000 nM T99089 CBL6M7 24879143 IC50 = 14000 nM T99089 CE74NO 24879204 IC50 = 12000 nM T99089 C48MIN 24879205 IC50 = 1200 nM T99089 CG5VC1 24879206 IC50 = 45000 nM T99089 CY18ZW 24879207 IC50 = 18000 nM T99089 C1XL8V 24879208 IC50 = 10000 nM T99089 C9SM2H 24879209 IC50 = 3800 nM T99089 CTPU27 24879260 IC50 = 76000 nM T99089 CBQN65 24879261 IC50 = 70000 nM T99089 CZ8CR2 24879262 IC50 = 45000 nM T99089 CD1QW9 24879263 IC50 = 36000 nM T99089 C8UPO4 24879264 IC50 = 5500 nM T99089 CDCN49 24879265 IC50 = 410 nM T99089 CYTM29 24879326 IC50 = 26000 nM T99089 C2F6KO 24879328 IC50 = 560 nM T99089 C6S2JM 24879329 IC50 > 100000 nM T99089 C1BJT3 24879330 IC50 = 22000 nM T99089 CK83CA 24879331 IC50 = 16000 nM T99089 C1CP0D 24879390 IC50 = 4700 nM T99089 CJZB61 24879392 IC50 = 19000 nM T99089 C8L0FE 24879393 IC50 = 31000 nM T99089 CT12IR 24879394 IC50 = 16000 nM T99089 C3T4CF 24879395 IC50 = 9800 nM T99089 CH4F5C 24879396 IC50 = 7400 nM T99089 C6TRZ7 24879462 IC50 = 44000 nM T99089 CKJ12G 24879463 IC50 = 1500 nM T99089 CGL5B4 24879464 IC50 = 29000 nM T99089 C4YA3G 24879465 IC50 = 29000 nM T99089 C96NEC 24879466 IC50 = 18000 nM T99089 CTZD56 24879467 IC50 = 22000 nM T99089 CAX20R 24879527 IC50 = 10000 nM T99089 CW8HQ4 24879528 IC50 = 56000 nM T99089 CBT3Y5 24879529 IC50 = 13000 nM T99089 C0ZBE3 24879530 IC50 = 19000 nM T99089 C7SQE5 24879531 IC50 = 34000 nM T99089 CV8Z3B 24879532 IC50 = 11000 nM T99089 C13QYB 24884503 IC50 = 24 nM T99089 C5E1YD 24891645 IC50 = 77 nM T99089 C2T9IQ 24891646 IC50 = 38 nM T99089 C4B7ND 24891647 IC50 = 57 nM T99089 C7Y8KZ 24891698 IC50 = 26.92 nM T99089 C6HE2Y 24891699 IC50 = 32 nM T99089 CK1R3B 24891700 IC50 = 51 nM T99089 CCY7G3 24891701 IC50 = 190 nM T99089 CJH19T 24894883 IC50 = 50000 nM T99089 CB5TP8 24894992 IC50 = 38000 nM T99089 CN13JF 24899915 IC50 = 0.74 ug.mL-1 T99089 CBWR97 24899916 IC50 = 1.5 ug.mL-1 T99089 C9F2JD 24899917 IC50 > 10 ug.mL-1 T99089 C64MTI 24900160 IC50 = 7.4 ug.mL-1 T99089 CO2I6Q 24900161 IC50 = 9 ug.mL-1 T99089 CQL3U0 24963235 IC50 = 1700 nM T99089 C26IGP 24963239 IC50 = 28 nM T99089 CJZE02 24963588 IC50 = 17 nM T99089 CAL45P 24963945 IC50 = 260 nM T99089 C1E7SQ 24964302 IC50 = 5 nM T99089 CA0QG4 24964658 IC50 = 6.5 nM T99089 C2U9TM 24965013 IC50 = 156 nM T99089 C09IXV 24965362 IC50 = 9 nM T99089 CR8N5G 24965367 IC50 = 1400 nM T99089 CTY2A7 24965371 IC50 = 41.5 nM T99089 C12PMT 24966065 IC50 = 18 nM T99089 CKRV37 24966066 IC50 = 15.4 nM T99089 C9YN2Q 24967131 IC50 = 42 nM T99089 COD0C3 24967871 IC50 = 216 nM T99089 CJ7ZD9 24968217 IC50 = 1500 nM T99089 C7HJU9 24968561 IC50 = 6.7 nM T99089 CT7S6C 24969040 IC50 = 360 nM T99089 CFDW17 24969041 IC50 > 10000 nM T99089 CD5HQ0 24969301 IC50 = 1540 nM T99089 C9NA3Z 24969303 IC50 > 10000 nM T99089 C9TQ4B 24969304 IC50 > 10000 nM T99089 C92TKX 24969393 IC50 = 1570 nM T99089 C78KAJ 24969394 IC50 > 10000 nM T99089 C97NFP 24969396 IC50 > 10000 nM T99089 C9FS1C 24969397 IC50 = 360 nM T99089 C85RQC 24969401 IC50 = 4270 nM T99089 CC23PA 24969484 IC50 > 10000 nM T99089 CDBL83 24969487 IC50 > 10000 nM T99089 CO4A0P 24969567 IC50 = 1030 nM T99089 CTJP28 24969568 IC50 > 10000 nM T99089 CL9UY3 24969569 IC50 > 10000 nM T99089 C0VK5E 24969668 IC50 = 500 nM T99089 CB9C5O 24969749 IC50 = 540 nM T99089 CW26KA 24969750 IC50 = 3600 nM T99089 C4AXL1 24969752 IC50 > 10000 nM T99089 CG6B9I 24969834 IC50 > 10000 nM T99089 C2M4FP 24969839 IC50 = 240 nM T99089 CB89UG 24969923 IC50 = 5880 nM T99089 C3K2VT 24970000 IC50 = 6340 nM T99089 CX8MC1 24970159 IC50 > 10000 nM T99089 CB0XA4 24970161 IC50 > 10000 nM T99089 CL7A6B 24970246 IC50 > 10000 nM T99089 C4G9WP 24986335 IC50 = 89 nM T99089 CDF57P 24995525 IC50 = 2.5 nM T99089 C9QO8R 25023945 IC50 = 57710 nM T99089 C4Y3FG 25023946 IC50 = 3750 nM T99089 CA61PS 25066845 IC50 = 22 nM T99089 CR46MG 25066846 IC50 = 2 nM T99089 C9Z3LB 25093294 IC50 = 86000 nM T99089 CM0E1C 25093324 IC50 = 68 nM T99089 CM4R0H 25093325 IC50 = 4.4 nM T99089 C5JX6H 25093326 IC50 = 1.5 nM T99089 C1DGE0 25093327 IC50 = 94 nM T99089 C9UW5V 25093328 IC50 = 70 nM T99089 C96EVA 25118036 IC50 = 51 nM T99089 CTV54O 25123227 IC50 > 10000 nM T99089 CG3XC9 25124150 IC50 = 80 nM T99089 CO2IR5 25124816 IC50 > 2000 nM T99089 C1IYN7 25127854 IC50 > 1000 nM T99089 CKD14B 25127856 IC50 = 290 nM T99089 CJBX60 25128180 IC50 > 1000 nM T99089 CC5SD9 25128181 IC50 > 1000 nM T99089 C9PL5S 25137959 IC50 > 25000 nM T99089 CVJ0S5 25137960 IC50 = 14 nM T99089 CJL80R 25161176 IC50 = 70 nM T99089 C85KCS 25178328 IC50 = 8000 nM T99089 CIG4H0 25178539 IC50 = 1200 nM T99089 C4GI6J 25178540 IC50 = 8400 nM T99089 CB6QT3 25195001 IC50 = 7 nM T99089 CYK1V8 25206185 IC50 = 5.6 nM T99089 C6FGQ1 25206346 IC50 = 47 nM T99089 C8ZBN0 25206349 IC50 = 15 nM T99089 CRO09K 25211064 IC50 = 8800 nM T99089 C41TLH 42603880 IC50 = 82000 nM T99089 CDM2N3 42606902 IC50 = 5940 nM T99089 CWS37O 42618140 IC50 > 10000 nM T99089 C2JV3O 42618143 IC50 > 10000 nM T99089 CG01BO 42618144 IC50 > 10000 nM T99089 CLD0M5 42625161 IC50 = 40 nM T99089 CS1CB9 42625162 IC50 = 85 nM T99089 CRUS43 42625163 IC50 > 100000 nM T99089 C27GYX 42625164 IC50 = 15900 nM T99089 CJ9EQ2 42625165 IC50 = 17200 nM T99089 CL8R1T 42625166 IC50 = 14000 nM T99089 C41PMY 42625241 IC50 = 28 nM T99089 CZPU80 42625242 IC50 > 100000 nM T99089 CDT39F 42625243 IC50 > 100000 nM T99089 CV5X0D 42625244 IC50 = 16700 nM T99089 C7HYW8 42625245 IC50 = 10000 nM T99089 CPV58O 42625246 IC50 > 100000 nM T99089 C3M2OV 42625324 IC50 = 10000 nM T99089 CC95QE 42625325 IC50 = 850 nM T99089 CV6CR3 42625326 IC50 > 100000 nM T99089 CK4Y8O 42625327 IC50 > 100000 nM T99089 CRP62O 42625328 IC50 > 100000 nM T99089 CIRG39 42625329 IC50 = 12200 nM T99089 CIR6N1 42625412 IC50 = 10000 nM T99089 C21YCQ 42625413 IC50 = 32500 nM T99089 CA1Y7G 42625505 IC50 = 23 nM T99089 CIGZ52 42626129 IC50 > 100000 nM T99089 CE6X4U 42626130 IC50 > 100000 nM T99089 C0IYC6 42626192 IC50 = 100 nM T99089 CMV35J 42626193 IC50 = 14 nM T99089 CN7A2L 42626194 IC50 > 100000 nM T99089 C98ZKU 42626195 IC50 > 100000 nM T99089 CP06XJ 42626196 IC50 = 21 nM T99089 C3GA4B 42626197 IC50 = 12 nM T99089 CWRD96 42626265 IC50 = 27 nM T99089 CLZ5T1 42626266 IC50 = 52 nM T99089 C4NW1Z 42626267 IC50 = 2840 nM T99089 CV3KQ7 42626268 IC50 = 600 nM T99089 C62UVE 42626269 IC50 = 860 nM T99089 CUA5H1 42626270 IC50 = 22 nM T99089 CEZW83 42626338 IC50 = 163 nM T99089 CQ9UV2 42626339 IC50 = 60 nM T99089 C5QG1C 42626340 IC50 = 46 nM T99089 CZ0CB6 42626341 IC50 = 61 nM T99089 CP2US6 42626342 IC50 = 305 nM T99089 CE2G9C 42626343 IC50 = 29 nM T99089 C4CX1E 42628843 IC50 = 5 nM T99089 CU9E4P 42629114 IC50 > 10000 nM T99089 CJ5U1X 42639664 IC50 = 6.5 ug.mL-1 T99089 CJT32G 42641056 IC50 = 600 nM T99089 CH8JQ9 42647197 IC50 = 464 nM T99089 CZP1I5 44131523 IC50 = 5 nM T99089 CRW8G5 44131524 IC50 = 4890 nM T99089 CYL5C1 44131526 IC50 = 168 nM T99089 CRN89T 44131527 IC50 = 187 nM T99089 CS15GI 44131710 IC50 = 4 nM T99089 C4LV1X 44131711 IC50 = 6 nM T99089 COH4S6 44131713 IC50 = 30 nM T99089 C7CJ9L 44132041 IC50 = 273 nM T99089 CLC25G 44132209 IC50 = 650 nM T99089 CZN36J 44132210 IC50 = 1080 nM T99089 CVEL46 44132212 IC50 = 222 nM T99089 CJ2U8W 44132374 IC50 = 43 nM T99089 CVC68Z 44132375 IC50 = 7 nM T99089 CN8D9W 44132531 IC50 = 134 nM T99089 CRAF54 44132532 IC50 = 280 nM T99089 CW8J5B 44132533 IC50 = 75 nM T99089 C1C0EF 44132534 IC50 = 640 nM T99089 C81MAW 44132690 IC50 = 7 nM T99089 C60THF 44132691 IC50 = 220 nM T99089 CKH43U 44132693 IC50 = 1700 nM T99089 CQB12C 44132694 IC50 = 8200 nM T99089 C7CH1O 44132849 IC50 = 600 nM T99089 CMIJ65 44132851 IC50 = 20 nM T99089 CF8IC2 44132852 IC50 = 101 nM T99089 C42STZ 44132853 IC50 = 15 nM T99089 C59VWU 44133012 IC50 = 2 nM T99089 CMG6E1 44133013 IC50 = 6 nM T99089 CL41OB 44133016 IC50 = 16000 nM T99089 C24APO 44133177 IC50 = 320 nM T99089 CW67CZ 44133180 IC50 = 3 nM T99089 C7OF9J 44133181 IC50 = 2 nM T99089 CIL5W6 44133361 IC50 = 750 nM T99089 CJK24I 44133362 IC50 = 3800 nM T99089 CVO95C 44133363 IC50 = 107 nM T99089 CM92WZ 44133364 IC50 = 246 nM T99089 C8TDB9 44133365 IC50 = 76 nM T99089 C1X4ZY 44133544 IC50 = 21 nM T99089 CZ20KG 44133545 IC50 = 390 nM T99089 CQ9M1C 44133546 IC50 = 133 nM T99089 CW8QC6 44133547 IC50 = 4200 nM T99089 CH9U7K 44133548 IC50 = 71 nM T99089 CZ0DA5 44133720 IC50 = 870 nM T99089 CMO9J8 44133721 IC50 = 7 nM T99089 CLSG50 44133722 IC50 = 21 nM T99089 CT6L2M 44133724 IC50 = 176 nM T99089 C94MCL 44133726 IC50 = 84 nM T99089 C4NDM9 44133727 IC50 = 108 nM T99089 CCSZ12 44133728 IC50 = 634 nM T99089 CV35ZJ 44133905 IC50 = 10 nM T99089 C97QTV 44133906 IC50 = 96 nM T99089 C3G4NP 44133907 IC50 = 10000 nM T99089 CI7OR1 44133908 IC50 = 8 nM T99089 CR2G0E 44133909 IC50 = 8 nM T99089 C4NP8V 44133910 IC50 = 105 nM T99089 CY1I5F 44133911 IC50 = 580 nM T99089 CTQ1A5 44133913 IC50 = 48 nM T99089 CZV39F 44133914 IC50 = 4 nM T99089 C5F6PH 44134083 IC50 = 80 nM T99089 C9WFA4 44134086 IC50 = 4 nM T99089 C7UIJ2 44134087 IC50 = 5 nM T99089 C8M2WR 44134089 IC50 = 3 nM T99089 CL0O7M 44134090 IC50 = 34 nM T99089 C4QOM5 44134091 IC50 = 306 nM T99089 CO42DC 44138048 IC50 > 10000 nM T99089 CL65QV 44138049 IC50 > 10000 nM T99089 CC9W0L 44185009 IC50 = 56 nM T99089 C1M8UL 44185010 IC50 = 22 nM T99089 CWT0K9 44185011 IC50 = 47 nM T99089 C2Q8MJ 44185012 IC50 = 37 nM T99089 CM4R5H 44185013 IC50 = 12 nM T99089 CAM26B 44185065 IC50 = 16 nM T99089 CW76EU 44185067 IC50 = 6 nM T99089 C2H5XO 44185068 IC50 = 37 nM T99089 CFTR94 44185069 IC50 = 220 nM T99089 C64GVD 44185123 IC50 = 1 nM T99089 CD04VP 44185124 IC50 = 25 nM T99089 C0YWR1 44185125 IC50 = 8 nM T99089 CVC9N0 44185126 IC50 = 106 nM T99089 CS5OR8 44185840 IC50 = 346 nM T99089 C3OZ0X 44185841 IC50 = 23 nM T99089 CRUD71 44185842 IC50 = 1060 nM T99089 C5GRD7 44185843 IC50 = 10 nM T99089 CJ15VW 44185844 IC50 = 3140 nM T99089 CVM46R 44185900 IC50 > 10000 nM T99089 C84DOE 44185901 IC50 = 5200 nM T99089 C12VEW 44185902 IC50 = 90 nM T99089 C3ZAK0 44185961 IC50 = 430 nM T99089 CL74HV 44186294 IC50 = 59000 nM T99089 CTB03L 44186295 IC50 = 559 nM T99089 CV6NG7 44186296 IC50 = 10000 nM T99089 C81UIO 44186297 IC50 = 6500 nM T99089 C9Q4XW 44186359 IC50 = 1330 nM T99089 CUTO28 44186360 IC50 = 1 nM T99089 CZEN24 44186361 IC50 = 12 nM T99089 C3PG7E 44186362 IC50 = 7 nM T99089 CVA0Z8 44186363 IC50 = 37 nM T99089 CY40HO 44186413 IC50 = 638 nM T99089 CEFN41 44186414 IC50 = 17 nM T99089 C3W8HZ 44186415 IC50 = 24 nM T99089 CS5OR3 44186416 IC50 = 167 nM T99089 CB5U6Q 44186417 IC50 > 100000 nM T99089 CSV05I 44186463 IC50 = 79 nM T99089 C7RQ3H 44186464 IC50 = 4600 nM T99089 CCFQ29 44187005 IC50 = 0.16 nM T99089 C6L0DV 44199408 IC50 = 38 nM T99089 CKJ29G 44199417 IC50 = 61 nM T99089 CN0D5T 44199425 IC50 = 17 nM T99089 C1X2HU 44199429 IC50 = 917 nM T99089 CMT07V 44207795 IC50 = 0.8 nM T99089 C6FKU5 44207796 IC50 = 1.6 nM T99089 CPHJ03 44207797 IC50 = 0.6 nM T99089 CPM2Y8 44217243 IC50 = 110 nM T99089 C0J7XH 44223152 IC50 = 14 nM T99089 CXNB60 44223174 IC50 = 2.2 nM T99089 CX7YO1 44223205 IC50 = 8.2 nM T99089 CD91HX 44223206 IC50 = 4.8 nM T99089 C5N4AB 44223207 IC50 = 1.8 nM T99089 CHA12Y 44223280 IC50 = 6.3 nM T99089 C9LHU2 44223282 IC50 = 19 nM T99089 C4CTE2 44223283 IC50 = 87 nM T99089 C6A7VR 44223334 IC50 = 6.2 nM T99089 C2Z8JX 44223468 IC50 = 7.5 nM T99089 CH0I7B 44223469 IC50 = 2.3 nM T99089 C42DBL 44223470 IC50 = 13 nM T99089 CF6U5Q 44223471 IC50 = 1.7 nM T99089 C1ZS2O 44223472 IC50 = 1.3 nM T99089 CDL87A 44223473 IC50 = 2.4 nM T99089 CG4EH1 44223627 IC50 = 32 nM T99089 CG74KN 44223631 IC50 = 2.4 nM T99089 C0XR3Z 44223650 IC50 = 4 nM T99089 CI8ZU0 44223675 IC50 = 1.1 nM T99089 CQ1N4G 44223692 IC50 = 12 nM T99089 CWCB51 44223693 IC50 = 2.7 nM T99089 CV6ZU8 44223890 IC50 = 9.2 nM T99089 CJ5Q7A 44223895 IC50 = 5.8 nM T99089 C8KT6W 44223912 IC50 = 3.4 nM T99089 C8KUI4 44223914 IC50 = 210 nM T99089 CM2T9S 44223915 IC50 = 88 nM T99089 CR7K2T 44223999 Ki = 1 nM T99089 CC38RW 44225585 IC50 = 87 nM T99089 CPRT47 44225586 IC50 = 1 nM T99089 CPH82M 44225587 IC50 = 4 nM T99089 C5SPW7 44225811 IC50 = 54.1 nM T99089 CF9OE0 44225812 IC50 < 2 nM T99089 CIP43R 44225813 IC50 = 0.4 nM T99089 C4JBC2 44225814 IC50 = 0.3 nM T99089 CR6SM1 44226026 IC50 = 8.5 nM T99089 CCT62X 44226027 IC50 = 43.5 nM T99089 CD29GR 44226028 IC50 = 0.5 nM T99089 C0UTL8 44226029 IC50 = 70.8 nM T99089 C89SFK 44226241 IC50 = 17 nM T99089 C7MB0L 44226447 IC50 = 0.9 nM T99089 CJUX24 44226448 IC50 = 9.7 nM T99089 CVT2A7 44226449 IC50 < 0.32 nM T99089 CA0C6B 44226657 IC50 = 3 nM T99089 CXM4N6 44227053 IC50 = 2 nM T99089 C8RDU2 44227055 IC50 = 0.4 nM T99089 C1CBY7 44227056 IC50 = 4.4 nM T99089 CF2BJ7 44227270 IC50 = 17 nM T99089 CJK49R 44227271 IC50 = 0.7 nM T99089 C2GHR8 44227272 IC50 = 4.4 nM T99089 CHX90P 44227273 IC50 = 45 nM T99089 CXD0P8 44227274 IC50 = 0.4 nM T99089 CC21ZI 44227474 IC50 > 1000 nM T99089 CI4CB1 44227477 IC50 > 1000 nM T99089 CZ37UW 44227694 IC50 = 46.6 nM T99089 CEL61X 44229839 IC50 > 10000 nM T99089 CY6C2X 44230849 IC50 = 1.6 nM T99089 CV7Q1M 44230852 IC50 = 40 nM T99089 CEW5F9 44230853 IC50 = 3.2 nM T99089 CK7LA1 44230854 IC50 = 1125 nM T99089 C7HC6Z 44230986 IC50 = 107 nM T99089 C4VL2B 44230987 IC50 = 167 nM T99089 CD5VW9 44230988 IC50 = 2.2 nM T99089 CJN28A 44230989 IC50 = 137 nM T99089 CR5C7A 44230990 IC50 = 4.4 nM T99089 C2Y8CF 44231119 IC50 = 1.5 nM T99089 CE5J4A 44231120 IC50 = 49 nM T99089 C0YE3K 44231121 IC50 = 2.2 nM T99089 C3T0VZ 44231122 IC50 = 1.1 nM T99089 C47HYD 44231123 IC50 = 86 nM T99089 CQW47T 44231243 IC50 = 1.4 nM T99089 C23DUC 44231244 IC50 = 1 nM T99089 CUJD31 44231246 IC50 = 8 nM T99089 C4ZV1S 44231247 IC50 = 0.76 nM T99089 C9GK4E 44231363 IC50 = 27 nM T99089 CC6B2Z 44231366 IC50 = 948 nM T99089 CDKW96 44231489 IC50 = 1560 nM T99089 C18YHD 44231490 IC50 = 60 nM T99089 CAKX67 44231491 IC50 = 59 nM T99089 CJW38K 44231605 IC50 = 31 nM T99089 CL2Q8X 44231720 IC50 = 1.4 nM T99089 C1JVN2 44231722 IC50 = 298 nM T99089 C41EIK 44231723 IC50 = 1.2 nM T99089 C2JU5V 44242890 IC50 = 93 nM T99089 CMO40X 44243006 IC50 = 2229 nM T99089 CDUE95 44243085 IC50 = 480 nM T99089 CI4DL6 44243129 IC50 = 121 nM T99089 CBG0P4 44243179 IC50 = 293 nM T99089 C8JVN0 44243219 IC50 = 52 nM T99089 CR30HI 44243260 IC50 = 165 nM T99089 C3EW0M 44243435 IC50 = 340 nM T99089 CT91HE 44243438 IC50 = 332 nM T99089 CTUV41 44243472 IC50 = 155 nM T99089 CA7NS4 44406429 IC50 = 13 nM T99089 CN3PH6 44406460 IC50 = 6 nM T99089 C43KQJ 44406537 IC50 = 12 nM T99089 CU09CR 44406595 IC50 = 1585 nM T99089 CC8Q4N 44406731 IC50 = 49600 nM T99089 C6B7KF 44406750 IC50 = 14000 nM T99089 CA5Q0P 44442388 IC50 = 34 nM T99089 C65YCN 44442389 IC50 = 138 nM T99089 CW02SD 44442390 IC50 = 175 nM T99089 C73GEP 44442391 IC50 = 6830 nM T99089 CX56BF 44442392 IC50 = 221 nM T99089 C6L3GV 44442393 IC50 = 1030 nM T99089 CX3J2I 44442394 IC50 = 397 nM T99089 C5QJ0P 44442395 IC50 = 634 nM T99089 CC3Z7Q 44442396 IC50 = 5 nM T99089 CLR10Z 44442397 IC50 = 110 nM T99089 C9UOK1 44442398 IC50 = 100 nM T99089 CE9T6W 44442399 IC50 = 153 nM T99089 CM6K2R 44442400 IC50 = 594 nM T99089 CW8JC5 44442401 IC50 = 349 nM T99089 CD1TY7 44442402 IC50 = 100 nM T99089 C4POG9 44442403 IC50 = 104 nM T99089 C0XHW1 44442404 IC50 = 112 nM T99089 CBSM51 44442405 IC50 = 156 nM T99089 CNT36H 44442406 IC50 = 142 nM T99089 CRA0Q8 44442407 IC50 = 165 nM T99089 C7YZ3M 44442408 IC50 = 101 nM T99089 CY9G0Q 44442409 IC50 = 146 nM T99089 C6XAR9 44442410 IC50 = 39 nM T99089 CJU4F6 44442411 IC50 = 64 nM T99089 CO0N1A 44442412 IC50 = 232 nM T99089 CIR9A7 44442413 IC50 = 192 nM T99089 CBQ51S 44442414 IC50 = 2560 nM T99089 CHP41T 44442415 IC50 = 191 nM T99089 CI26UX 44442416 IC50 = 154 nM T99089 C2W1RN 44442417 IC50 = 122 nM T99089 C4A9FD 44442418 IC50 = 69 nM T99089 CKC3J0 44442419 IC50 = 40 nM T99089 C10MKH 44448311 IC50 = 274 nM T99089 C1QN4V 44448333 IC50 = 141 nM T99089 CLQF97 44448334 IC50 = 469 nM T99089 C73THQ 44448354 IC50 = 16 nM T99089 C8XOE9 44448666 IC50 = 10 nM T99089 CEOA67 44448669 IC50 = 83 nM T99089 C0DPU3 44448725 IC50 = 18 nM T99089 CFQN07 44448726 IC50 = 85 nM T99089 CR85LO 44448746 IC50 = 40 nM T99089 C5Y2JR 44448747 IC50 = 3 nM T99089 CA76JX 44448748 IC50 = 4 nM T99089 C7N2AQ 44473101 IC50 = 34 nM T99089 C4MG3F 44473102 IC50 = 56 nM T99089 CA85NJ 44473103 IC50 = 44 nM T99089 C6Q7NU 44479258 IC50 = 2120 nM T99089 C29ZDL 44479262 IC50 = 23740 nM T99089 C0Y5OQ 44479517 IC50 = 2740 nM T99089 C3VRO9 44557921 IC50 > 10000 nM T99089 CVLW62 44569182 IC50 > 100000 nM T99089 CFQ6C8 44569219 IC50 > 100000 nM T99089 C1QLZ3 44571660 IC50 = 5 nM T99089 CDW02V 44571710 IC50 = 10500 nM T99089 C1L7TV 44571711 IC50 = 1 nM T99089 CT4DF8 44571712 IC50 = 21100 nM T99089 CJ69GM 44571753 IC50 = 580 nM T99089 CY0I9Q 44571754 IC50 = 1200 nM T99089 C4EHC9 44571755 IC50 = 625 nM T99089 CI8V0L 44571800 IC50 = 322 nM T99089 C7S0LB 44571801 IC50 = 16 nM T99089 CVJU90 44571802 IC50 = 15 nM T99089 C85RJP 44571803 IC50 = 16 nM T99089 CWFB42 44571820 IC50 = 320 nM T99089 CTRD67 44571867 IC50 = 15 nM T99089 CWN95Q 44571868 IC50 = 28 nM T99089 CQ09OS 44571869 IC50 = 237 nM T99089 C7M0ET 44571870 IC50 = 11 nM T99089 CTM2J1 44571913 IC50 = 30 nM T99089 C58MVO 44571914 IC50 = 115 nM T99089 CX5GH1 44571915 IC50 = 9 nM T99089 C21DSM 44571916 IC50 = 14 nM T99089 CWP80I 44571963 IC50 = 48 nM T99089 CGIH39 44571964 IC50 = 116 nM T99089 CCM0D8 44571965 IC50 = 38 nM T99089 C0M7TJ 44571966 IC50 = 79 nM T99089 CV17DO 44572009 IC50 = 48 nM T99089 C03AOY 44572010 IC50 = 205 nM T99089 CLG7X2 44572011 IC50 = 16 nM T99089 C9IPZ6 44572058 IC50 = 35 nM T99089 C42XRK 44572059 IC50 = 17 nM T99089 CDRK26 44572109 IC50 = 76 nM T99089 CP04MY 44583650 IC50 = 7 nM T99089 CM2RZ1 44586991 IC50 = 0.57 nM T99089 CFHM64 44587046 IC50 = 3.91 nM T99089 CW9KM4 44587047 IC50 = 0.04 nM T99089 C1MH9X 44587048 IC50 = 0.09 nM T99089 CFL31E 44587049 IC50 = 1.16 nM T99089 CMKX28 44587190 IC50 = 0.05 nM T99089 CY4V5F 44587191 IC50 = 0.56 nM T99089 C8KCO7 44587210 IC50 = 4.02 nM T99089 CTH20X 44587211 IC50 = 0.47 nM T99089 CU8E5Z 44587234 IC50 = 0.85 nM T99089 CXQ8E3 44587235 IC50 = 0.23 nM T99089 C9O4LW 44587236 IC50 = 969.6 nM T99089 C5FW7T 44587271 IC50 = 433.8 nM T99089 C3MO4A 44587272 IC50 = 68.4 nM T99089 CR3VE4 44587273 IC50 = 4.1 nM T99089 CI1K9L 44587274 IC50 = 2.1 nM T99089 CRZ43D 44587295 IC50 = 2.9 nM T99089 CY09FE 44587296 IC50 = 3.1 nM T99089 CWU29I 44587510 IC50 = 331 nM T99089 CNU73X 44587528 IC50 = 41.7 nM T99089 C8O3ES 44587529 IC50 = 170 nM T99089 C58DLS 44587530 IC50 = 110 nM T99089 C5QXC0 44587531 IC50 = 5.3 nM T99089 C5R2EI 44587550 IC50 = 25.7 nM T99089 CQN15G 44587551 IC50 = 10.5 nM T99089 C7OI4S 44587552 IC50 = 3.9 nM T99089 CM0UX7 44587582 IC50 = 5.4 nM T99089 CCS62T 44587583 IC50 = 2.1 nM T99089 CB4O9Z 44587584 IC50 = 79.4 nM T99089 C3Y5AW 44589519 IC50 = 7 nM T99089 C09EWJ 44590206 IC50 = 31 nM T99089 C3LZ6B 44593434 IC50 = 49 nM T99089 C7BX3O 44602984 IC50 = 80 nM T99089 C86VZL 44602985 IC50 = 67 nM T99089 C8KI5C 44603044 IC50 = 24000 nM T99089 C4M2KB 44654329 IC50 = 190 nM T99089 CGX7Q4 45267129 IC50 = 1450 nM T99089 C4GRT3 45267957 IC50 > 10000 nM T99089 C65XTQ 45267989 IC50 > 10000 nM T99089 C0DN8Q 45268879 IC50 = 7070 nM T99089 C3VI6H 45268883 IC50 = 170 nM T99089 CF17WS 45269730 IC50 = 160 nM T99089 CCZ72A 45271358 IC50 > 10000 nM T99089 C17RYH 45271371 IC50 = 410 nM T99089 C8L9ZU 45273140 IC50 = 270 nM T99089 CWI2D1 45375869 IC50 = 30 nM T99089 C2D6QS 45486182 IC50 < 2 nM T99089 C82YQR 45486184 IC50 = 9.1 nM T99089 CLMF90 45486187 IC50 = 3.8 nM T99089 C76ENX 45486190 IC50 < 0.3 nM T99089 CE1MZ4 45486203 IC50 = 302 nM T99089 CR6E9Y 45486205 IC50 = 22.8 nM T99089 C28GPA 45486206 IC50 = 39.4 nM T99089 CO81AX 45486208 IC50 = 151 nM T99089 C4V1FW 45486210 IC50 = 2.1 nM T99089 CPO7F8 45486211 IC50 = 4.9 nM T99089 C6EX1G 45486212 IC50 = 8.4 nM T99089 CDK4T2 45486218 IC50 = 57.9 nM T99089 COI1M7 45486219 IC50 = 36 nM T99089 CVJ34H 45486222 IC50 > 1000 nM T99089 CEQ4O7 45486223 IC50 = 6.4 nM T99089 CVK3E8 45486224 IC50 = 67 nM T99089 CB6L4I 45486225 IC50 = 6.7 nM T99089 CQ8J5U 45486226 IC50 = 75.9 nM T99089 C4UF0V 45503363 IC50 = 140 nM T99089 CYQ8B2 45503364 IC50 = 190 nM T99089 C32HLA 45503367 IC50 = 140 nM T99089 C2KZ8V 46196674 IC50 = 27 nM T99089 CV4GE7 46196675 IC50 = 70 nM T99089 CI84VY 46196676 IC50 = 75 nM T99089 CT1P2W 46196677 IC50 = 40 nM T99089 CG2AU5 46196996 IC50 = 62 nM T99089 C38BVC 46196997 IC50 = 122 nM T99089 CCL6H2 46196998 IC50 = 52 nM T99089 CF3GQ1 46196999 IC50 = 76 nM T99089 CO9ML6 46197110 IC50 = 70 nM T99089 CW3ZC7 46197111 IC50 = 2200 nM T99089 CXYD95 46197658 IC50 = 83 nM T99089 C61LOS 46197659 IC50 = 1190 nM T99089 C2U6BA 46197660 IC50 = 147 nM T99089 CRU91A 46197661 IC50 = 210 nM T99089 C1UN6H 46197662 IC50 = 104 nM T99089 C15SIF 46197769 IC50 = 28000 nM T99089 CV7B0P 46197770 IC50 = 124 nM T99089 C2C6OJ 46197771 IC50 = 140 nM T99089 CJB83Y 46197772 IC50 = 70000 nM T99089 CL5Q6E 46197773 IC50 = 620 nM T99089 CD1B2I 46197872 IC50 = 42 nM T99089 CCOB85 46197873 IC50 = 142 nM T99089 C5WPQ2 46197874 IC50 = 7800 nM T99089 COSG68 46197875 IC50 = 170 nM T99089 CC1OD0 46197876 IC50 = 84 nM T99089 C7S9KB 46197980 IC50 = 176 nM T99089 C4D1FE 46197981 IC50 = 143 nM T99089 CH5ZX1 46197982 IC50 = 164 nM T99089 CKD01G 46197983 IC50 = 830 nM T99089 C6Y7NW 46197984 IC50 = 90 nM T99089 CIJ2C6 46198095 IC50 = 2900 nM T99089 C3OJS6 46198096 IC50 = 130 nM T99089 CM37LV 46198097 IC50 = 54 nM T99089 C32EMV 46198098 IC50 = 36 nM T99089 C6FK0L 46198099 IC50 = 190 nM T99089 CS8P1X 46198205 IC50 = 240 nM T99089 C6OQH7 46198206 IC50 = 11 nM T99089 C2XF3D 46198207 IC50 = 510 nM T99089 COX8S7 46198208 IC50 = 14 nM T99089 C5CP2F 46198209 IC50 = 35 nM T99089 CQ1D4O 46198316 IC50 = 251 nM T99089 CGU80Q 46198317 IC50 = 100 nM T99089 CM58LS 46198318 IC50 = 383 nM T99089 CL7UY0 46198320 IC50 = 197 nM T99089 CBO87C 46198375 IC50 < 0.32 nM T99089 CUA97D 46209401 IC50 = 2 nM T99089 CMBJ68 46222580 IC50 = 26 nM T99089 C1GO2Y 46222581 IC50 = 360 nM T99089 CR2G0M 46228457 IC50 = 26 nM T99089 CRQ0V5 46228458 IC50 = 195 nM T99089 CIV52B 46228459 IC50 = 740 nM T99089 CCF60G 46228460 IC50 = 128 nM T99089 C2P9QO 46228508 IC50 = 89 nM T99089 CH8M7J 46228509 IC50 = 123 nM T99089 C2Q5RG 46228510 IC50 = 400 nM T99089 CUY82H 46228511 IC50 = 21300 nM T99089 CZ76CV 46228524 IC50 = 17800 nM T99089 CCF84Y 46228525 IC50 = 730 nM T99089 CW96RT 46228526 IC50 = 690 nM T99089 CCO78J 46228527 IC50 = 620 nM T99089 CQKD47 46228552 IC50 = 87000 nM T99089 C82CNS 46228553 IC50 = 94000 nM T99089 CXV41S 46228554 IC50 = 68000 nM T99089 C59GQX 46228555 IC50 = 42000 nM T99089 CJ1V9Y 46228556 IC50 = 14 nM T99089 C8J4GN 46228587 IC50 > 10000 nM T99089 CZR4K2 46228588 IC50 = 79000 nM T99089 CXE9G2 46228589 IC50 = 49 nM T99089 CK07MJ 46228590 IC50 = 6700 nM T99089 C9TW1K 46228617 IC50 = 15000 nM T99089 CJ0M5L 46228618 IC50 = 71 nM T99089 CZ7AI8 46228619 IC50 = 23 nM T99089 CG10QD 46228620 IC50 = 6480 nM T99089 CGE71D 46228640 IC50 = 17 nM T99089 C1BZ8D 46228641 IC50 = 40 nM T99089 C4IJ0T 46228642 IC50 = 57 nM T99089 CHS4I6 46228643 IC50 > 10000 nM T99089 CRX8M3 46228664 IC50 = 115 nM T99089 C94GNC 46228665 IC50 = 15400 nM T99089 CK9HB1 46228666 IC50 = 920 nM T99089 CN1SB2 46228667 IC50 > 100000 nM T99089 C6RNZ2 46228694 IC50 > 100000 nM T99089 CYJG41 46228695 IC50 = 22000 nM T99089 C9J3EO 46228696 IC50 > 100000 nM T99089 CLJ4Z0 46228697 IC50 = 93000 nM T99089 C1KG2A 46228728 IC50 = 1000 nM T99089 CVI1J2 46228729 IC50 = 79000 nM T99089 CKX81Z 46228730 IC50 = 92000 nM T99089 C7NFH5 46228731 IC50 > 100000 nM T99089 C8XB1I 46228766 IC50 = 38000 nM T99089 C3YT8B 46228767 IC50 = 13700 nM T99089 CPA46C 46228768 IC50 = 87 nM T99089 CH0ES4 46228769 IC50 = 48 nM T99089 C2B5ES 46228792 IC50 = 15 nM T99089 C0NP5I 46228793 IC50 = 23 nM T99089 C9NRH2 46228794 IC50 = 6800 nM T99089 COW38I 46228795 IC50 = 90 nM T99089 CR0EO8 46228796 IC50 = 4700 nM T99089 C1Z4XW 46228797 IC50 = 8000 nM T99089 CA4M3D 46228798 IC50 = 187 nM T99089 C8CX5F 46228818 IC50 > 100000 nM T99089 C9EMG4 46228819 IC50 = 57000 nM T99089 CCG2J8 46228820 IC50 > 100000 nM T99089 C8ZO7J 46228821 IC50 = 11300 nM T99089 C6E5PY 46228822 IC50 = 356 nM T99089 C07ZPY 46228823 IC50 = 590 nM T99089 COW7Q6 46228824 IC50 = 500 nM T99089 C6L0JY 46228825 IC50 > 10000 nM T99089 CLS64M 46228853 IC50 > 100000 nM T99089 CH82DK 46228854 IC50 = 1660 nM T99089 CH65DP 46228855 IC50 = 850 nM T99089 CJ85WB 46228856 IC50 = 124 nM T99089 CE60UA 46228857 IC50 > 100000 nM T99089 CC0AT1 46228858 IC50 > 10000 nM T99089 CAE8F0 46228859 IC50 > 10000 nM T99089 C5QU9B 46228860 IC50 = 240 nM T99089 CJZA13 46228900 IC50 = 15900 nM T99089 C8KNZ9 46228901 IC50 = 1560 nM T99089 CPY3I0 46228902 IC50 = 14000 nM T99089 CQ8V3N 46228903 IC50 = 25200 nM T99089 C3EBU0 46228904 IC50 > 100000 nM T99089 C68LVX 46228905 IC50 = 770 nM T99089 C5JZF2 46228906 IC50 = 33 nM T99089 CX0J3H 46228907 IC50 = 340 nM T99089 CZM90S 46228908 IC50 = 64 nM T99089 CJ9EI6 46228945 IC50 = 21100 nM T99089 C4F7IE 46228946 IC50 > 100000 nM T99089 C6N2SC 46228947 IC50 = 2750 nM T99089 C48RIK 46228948 IC50 = 1120 nM T99089 CI9WF8 46228949 IC50 = 33 nM T99089 CYP51A 46228950 IC50 = 6900 nM T99089 C3T8AM 46228951 IC50 = 7 nM T99089 CIM53K 46847263 IC50 = 1.7 nM T99089 C7H4YM 46865419 IC50 = 80 nM T99089 C4MKC5 46870033 IC50 = 17 nM T99089 CJMO86 46879449 IC50 = 0.51 nM T99089 C4KQ3H 46879450 IC50 = 0.5 nM T99089 CNH1L4 46879451 IC50 = 12 nM T99089 C8FC5Y 46879452 IC50 = 0.44 nM T99089 C6Z1XG 46879458 IC50 = 42 nM T99089 CIY3O5 46879459 IC50 = 98 nM T99089 C75CRZ 46879460 IC50 = 18 nM T99089 CT6QA4 46879461 IC50 = 30 nM T99089 CV03IY 46879517 IC50 = 8.7 nM T99089 CSO84N 46879518 IC50 = 8.2 nM T99089 CF1BT0 46879519 IC50 = 21 nM T99089 CBRS82 46879520 IC50 = 1 nM T99089 CK7LQ4 46879877 IC50 = 552 nM T99089 C79IHJ 46879959 IC50 = 842 nM T99089 C9XLF4 46879960 IC50 = 308 nM T99089 CQ25VN 46879961 IC50 > 10000 nM T99089 CZ6D2P 46880014 IC50 = 2 nM T99089 C09EYD 46880015 IC50 = 1.5 nM T99089 CMO47N 46880016 IC50 = 57 nM T99089 C2WA7P 46880017 IC50 = 139 nM T99089 CXTC97 46880018 IC50 = 34 nM T99089 C2DUH7 46880019 IC50 = 40 nM T99089 CGQ93K 46880020 IC50 = 318 nM T99089 CSD1Q7 46880021 IC50 = 41 nM T99089 C0G1KP 46880074 IC50 = 1 nM T99089 CB14IR 46880075 IC50 = 0.49 nM T99089 C5WD3A 46880076 IC50 < 0.32 nM T99089 C0F9VH 46880077 IC50 = 26 nM T99089 C6NGU8 46880078 IC50 = 117 nM T99089 CQT06S 46880079 IC50 = 44 nM T99089 CZYQ96 46880102 IC50 < 0.32 nM T99089 CI72BX 46880103 IC50 < 0.32 nM T99089 C7SK8G 46880104 IC50 < 0.32 nM T99089 CAFD60 46880105 IC50 = 20 nM T99089 COA93M 46880106 IC50 = 38 nM T99089 CF24RO 46880107 IC50 = 113 nM T99089 CJOM49 46880136 IC50 = 0.38 nM T99089 C7ZMV0 46880137 IC50 < 0.32 nM T99089 CQY7E2 46880138 IC50 < 0.32 nM T99089 C4V3UA 46880139 IC50 = 112 nM T99089 CHZL13 46880140 IC50 = 44 nM T99089 CL0W5N 46880141 IC50 = 941 nM T99089 CWL70U 46880217 IC50 < 0.32 nM T99089 C9AZE3 46880218 IC50 < 0.32 nM T99089 C4MT6A 46880225 IC50 = 84 nM T99089 CKXA51 46880226 IC50 = 393 nM T99089 C5YQC6 46880227 IC50 = 326 nM T99089 C0V6PO 46880228 IC50 = 362 nM T99089 C38CFM 46880229 IC50 = 219 nM T99089 C0NT9Z 46883533 IC50 > 10000 nM T99089 C1G4BN 46883535 IC50 > 10000 nM T99089 C12VIL 46883538 IC50 > 10000 nM T99089 CV28UF 46883539 IC50 = 100 nM T99089 CS4VH0 46883569 IC50 > 10000 nM T99089 C6M5GU 46883570 IC50 = 6200 nM T99089 CC1I3F 46883571 IC50 > 10000 nM T99089 C16TPN 46883708 IC50 = 1100 nM T99089 C3AVB1 46883709 IC50 = 4000 nM T99089 CZ8XB2 46883710 IC50 = 660 nM T99089 CMR2G9 46883711 IC50 = 60 nM T99089 CL0ZT3 46883714 IC50 = 25 nM T99089 CQ4X5O 46883715 IC50 = 40 nM T99089 C9EL2F 46883716 IC50 = 53 nM T99089 CG0VM7 46883717 IC50 = 160 nM T99089 C1N6OV 46883718 IC50 = 130 nM T99089 CZB28E 46883719 IC50 = 68 nM T99089 C4PS8I 46883720 IC50 = 110 nM T99089 CEH9Q2 46883721 IC50 = 110 nM T99089 C5PD6F 46883722 IC50 = 66 nM T99089 CPF9D2 46883723 IC50 = 66 nM T99089 CV42XD 46885361 IC50 > 10000 nM T99089 C9TME7 46885362 IC50 = 540 nM T99089 C0P7GZ 46885363 IC50 = 1110 nM T99089 CQ0ZK1 46885411 IC50 > 10000 nM T99089 C9XB7U 46885412 IC50 > 10000 nM T99089 CGYW52 46885477 IC50 > 10000 nM T99089 COJA32 46892971 IC50 = 1200 nM T99089 C7E9SF 46899944 IC50 = 17 nM T99089 C5T4OX 46899945 IC50 = 64 nM T99089 C4UG0X 46899948 IC50 = 258 nM T99089 CC0A1B 46900109 IC50 = 59 nM T99089 CPCD05 46900110 IC50 = 141 nM T99089 CJ5L9R 46900111 IC50 = 405 nM T99089 C20YBF 46900112 IC50 = 69 nM T99089 CVS9U2 46900113 IC50 = 42 nM T99089 CCBO60 46900264 IC50 = 17 nM T99089 C16LWK 46900265 IC50 = 25 nM T99089 C1I6HG 46900266 IC50 = 730 nM T99089 CP45QN 46900267 IC50 = 1670 nM T99089 CAOI74 46900268 IC50 = 1370 nM T99089 CFNK12 46900424 IC50 = 55 nM T99089 CK7T2S 46900425 IC50 = 58 nM T99089 C10CRA 46900426 IC50 = 87 nM T99089 C0Z9PF 46900427 IC50 = 69 nM T99089 CCV9L5 46900428 IC50 = 51 nM T99089 CQR3A5 46901756 IC50 = 5 nM T99089 CZ7M4V 46919120 IC50 = 180.1 nM T99089 C5WBZ7 46919121 IC50 < 1 nM T99089 CNL40R 46919122 IC50 = 413.9 nM T99089 CWGT04 46919517 IC50 = 9.1 nM T99089 CP59KI 46919518 IC50 = 15 nM T99089 C9E4YG 46919605 IC50 = 2 nM T99089 C9Z2QG 46919606 IC50 = 3 nM T99089 C9O0AN 46927521 EC50 = 9 nM T99089 C1L2PQ 46927522 EC50 = 4 nM T99089 C6OJA1 46927597 EC50 = 7 nM T99089 C9PAT7 46927672 IC50 = 3.8 nM T99089 CSOG58 46937280 IC50 = 240 nM T99089 C02IJE 46937281 IC50 = 230 nM T99089 C7LK1C 46945257 IC50 = 19500 nM T99089 CHX76J 49784892 IC50 > 1000 nM T99089 CA1H8S 49784893 IC50 > 1000 nM T99089 CTZG05 49784988 IC50 > 1000 nM T99089 CG2IO7 49785079 IC50 > 1000 nM T99089 CZI34V 49785167 IC50 > 1000 nM T99089 CJK65T 49785253 IC50 > 1000 nM T99089 C3NV0J 49785827 IC50 > 1000 nM T99089 C1AR4G 49785829 IC50 > 1000 nM T99089 CR9WA4 49836427 IC50 = 0.51 nM T99089 CX1ZO4 49836539 IC50 = 0.23 nM T99089 C7F8JO 49836540 IC50 < 0.1 nM T99089 C0X2FY 49836541 IC50 < 0.32 nM T99089 C82UYD 49836542 IC50 = 1.4 nM T99089 CL1CV3 49836646 IC50 = 7.3 nM T99089 C9V1JH 49836647 IC50 = 1.9 nM T99089 C1G8OB 49836648 IC50 = 2 nM T99089 CU3KH0 49836649 IC50 = 1 nM T99089 CWTL58 49836748 IC50 = 0.61 nM T99089 CJX81B 49836749 IC50 = 0.38 nM T99089 CDXE39 49836750 IC50 = 9.6 nM T99089 COYU08 49836854 IC50 = 0.35 nM T99089 C2RO1T 49836856 IC50 = 61 nM T99089 CFX3P6 49836857 IC50 = 0.5 nM T99089 C5R6HU 49836964 IC50 < 0.32 nM T99089 CXW48M 49836965 IC50 < 0.1 nM T99089 CO3K1E 49836966 IC50 = 0.11 nM T99089 C1AZW5 49836968 IC50 = 0.71 nM T99089 CTC01J 49837087 IC50 = 0.41 nM T99089 CD1XZ0 49837088 IC50 = 10 nM T99089 CGO4Q1 49837089 IC50 = 1.2 nM T99089 CUM13L 49837090 IC50 = 0.52 nM T99089 C5H0XP 49837198 IC50 = 0.77 nM T99089 CGO6B2 49837300 IC50 < 0.32 nM T99089 CTH0Z6 49837301 IC50 < 0.32 nM T99089 CNA43S 49837401 IC50 < 0.32 nM T99089 CSI9D6 49837402 IC50 < 0.32 nM T99089 CN89TG 49840317 IC50 > 15000 nM T99089 CY48DE 49849970 IC50 = 1.4 nM T99089 CUS56N 49863686 IC50 > 100000 nM T99089 CIU7C1 49863687 IC50 > 100000 nM T99089 CHL4D9 49863710 IC50 > 100000 nM T99089 CUCO48 49863711 IC50 = 92.3 nM T99089 CCPS95 49863903 IC50 = 54 nM T99089 CZIR49 49863968 IC50 = 6600 nM T99089 CMJ70C 50912930 IC50 = 0.54 nM T99089 CS7J8G 50937465 IC50 = 2.9 nM T99089 C36LQJ 50940491 IC50 = 4 nM T99089 C2Q0GE 50990922 IC50 = 3 nM T99089 CT7UB5 50990960 IC50 = 7 nM T99089 C61DVY 50990961 IC50 = 2.7 nM T99089 CV3UP9 50992247 IC50 = 2.1 nM T99089 CSW27B 50994972 IC50 = 374 nM T99089 CYNX05 50994975 IC50 = 129 nM T99089 C4XV7W 50994976 IC50 = 174 nM T99089 CE73LF 50994977 IC50 = 190 nM T99089 C53WVZ 50995007 IC50 = 83.18 nM T99089 C8OWU5 50995160 IC50 = 367 nM T99089 CZ4B5Q 50995530 IC50 = 0.9 nM T99089 CMR62F 50995532 IC50 = 1.096 nM T99089 CD7KN6 50995705 EC50 = 2.6 nM T99089 CRJL51 50995706 IC50 = 5.6 nM T99089 CRB3V5 50995710 IC50 = 3.2 nM T99089 C59ESV 50996310 IC50 = 1.8 nM T99089 CL7FA8 50997340 IC50 = 36 nM T99089 C63VKR 50997526 IC50 = 141.25 nM T99089 CWN50H 50997675 IC50 = 43 nM T99089 CLIK35 50997676 IC50 = 247 nM T99089 CBQU14 50997677 IC50 = 299 nM T99089 COC1I5 50997678 IC50 = 228 nM T99089 CTMF09 50997679 IC50 = 128 nM T99089 CWN54R 51003389 IC50 = 4.2 nM T99089 C5OUV8 51003390 IC50 = 240 nM T99089 C5X9OM 51354603 IC50 = 61 nM T99089 C4DSG2 51354885 IC50 = 8 nM T99089 CQ85FC 51354886 IC50 = 3.3 nM T99089 C7MOQ0 51354887 IC50 = 2.9 nM T99089 C5KVT1 51355181 IC50 = 5 nM T99089 CS5F4Z 51355182 IC50 = 6 nM T99089 C4NFL7 51355183 IC50 = 4 nM T99089 C4W6PY 51355459 IC50 = 5 nM T99089 C95FWU 51355461 IC50 = 2.2 nM T99089 C4J3RE 51355733 IC50 = 7 nM T99089 C7LO2Y 52932687 IC50 = 630 nM T99089 C6DKQ4 52932689 IC50 = 100 nM T99089 C87LMF 52932691 IC50 = 32000 nM T99089 CNW01S 52932692 IC50 = 1300 nM T99089 C7XI4R 52932914 IC50 = 160 nM T99089 C8FBT0 52932915 IC50 = 800 nM T99089 CBVW62 52932917 IC50 = 2500 nM T99089 C7XVM5 52933152 IC50 = 1000 nM T99089 C1L6UP 52933587 IC50 = 40 nM T99089 CG04VW 52933647 IC50 = 79 nM T99089 C4L8GI 52934106 IC50 = 50 nM T99089 C9UYP8 52934570 IC50 = 130 nM T99089 CE8L9U 52934573 IC50 = 1000 nM T99089 CL16MA 52934795 IC50 = 400 nM T99089 C91KNR 52934796 IC50 = 250 nM T99089 CQ2ET7 52935028 IC50 = 10000 nM T99089 CJ1E7O 52935890 IC50 = 79 nM T99089 CD1XK2 52936114 IC50 = 1000 nM T99089 CK12ZP 52936117 IC50 = 4000 nM T99089 C4DLK1 52941323 IC50 = 4400 nM T99089 C02RNH 52941410 IC50 = 730 nM T99089 CKWC23 52942546 IC50 = 1330 nM T99089 CVE49F 52943666 IC50 > 10000 nM T99089 CI4Z7O 52943694 IC50 = 1710 nM T99089 C43TJA 52944042 IC50 = 970 nM T99089 C9MV6T 52945093 IC50 > 10000 nM T99089 CD9G0Y 52945288 IC50 = 1200 nM T99089 CG0BA4 52946221 IC50 = 740 nM T99089 CN8X0H 52947491 IC50 = 840 nM T99089 CDV8T6 52948574 IC50 = 3700 nM T99089 CWY5V9 52948575 IC50 = 1840 nM T99089 CUZ65L 52948582 IC50 > 10000 nM T99089 C4Q9IX 52948946 IC50 = 1600 nM T99089 CQ6IB5 52949635 IC50 = 1.2 nM T99089 CPM59C 52950212 IC50 = 1.4 nM T99089 C1SKV3 53249125 EC50 = 2100 nM T99089 CFRH86 53302367 IC50 = 1.6 nM T99089 CEZ7P6 53313343 IC50 = 1.6 nM T99089 CNKP63 53316555 IC50 = 1400 nM T99089 CN3Y4C 53316581 IC50 = 5 nM T99089 CDX1O6 53316582 IC50 = 2 nM T99089 C65DAZ 53316583 IC50 < 2 nM T99089 C3LTA4 53317522 IC50 = 93 nM T99089 C87OAQ 53317986 IC50 = 0.8 nM T99089 CE1V5K 53319219 IC50 = 3 nM T99089 CM0N2P 53319337 IC50 = 5.2 nM T99089 C7XI0Q 53319338 IC50 = 179 nM T99089 C1L8WR 53319339 IC50 = 2.4 nM T99089 CFN2J5 53320305 IC50 = 5800 nM T99089 CIOP36 53320502 IC50 = 1200 nM T99089 CC2IW7 53320600 IC50 = 4.3 nM T99089 CN1TI4 53320630 IC50 = 38 nM T99089 CZN0B8 53320631 IC50 = 0.3 nM T99089 CMQI43 53321817 IC50 = 570 nM T99089 CW7B3H 53321844 IC50 = 1500 nM T99089 C92UFO 53321929 IC50 = 5 nM T99089 CY0V2M 53323287 IC50 = 14 nM T99089 C4HKE1 53323288 IC50 = 5.7 nM T99089 CA4T3Y 53323289 IC50 = 2.7 nM T99089 CNW02P 53323290 IC50 = 0.8 nM T99089 CP41WD 53324073 IC50 = 4 nM T99089 CJ4G3Y 53324074 IC50 = 2 nM T99089 C62GPL 53324318 IC50 = 8200 nM T99089 CL4G1V 53324616 IC50 = 30 nM T99089 CNO54Z 53324617 IC50 = 2.3 nM T99089 CFP84X 53324920 IC50 = 3.2 nM T99089 CBY49I 53325802 IC50 = 32 nM T99089 CD9O2F 53325830 IC50 < 2 nM T99089 C1EXW0 53325922 IC50 = 2 nM T99089 C2JB0Z 53325923 IC50 = 1.6 nM T99089 CCK30V 53379548 IC50 = 2490 nM T99089 C48TNF 53379553 IC50 = 59110 nM T99089 CCTS15 53380119 IC50 = 9070 nM T99089 CGVD50 53380120 IC50 = 13540 nM T99089 C5S1UJ 53380121 IC50 = 3760 nM T99089 CHK92L 53380218 IC50 = 22650 nM T99089 CF7U6Q 53380219 IC50 = 45090 nM T99089 CD19RY 53380221 IC50 = 28510 nM T99089 C4SWC9 53380318 IC50 = 21990 nM T99089 CZ3OU5 53380319 IC50 = 20500 nM T99089 CF9JU3 53380320 IC50 = 91550 nM T99089 CK21TC 53380322 IC50 = 1620 nM T99089 CC1D5H 53380323 IC50 = 2810 nM T99089 C4GB3K 53380324 IC50 = 8890 nM T99089 CVG90B 53389651 IC50 > 10000 nM T99089 C3HMP1 53484099 IC50 = 8.6 nM T99089 CTGC73 54580078 IC50 = 3800 nM T99089 CL5Q6F 54580136 IC50 = 8 nM T99089 CQOT43 54580519 IC50 = 7 nM T99089 C89YCL 54580728 EC50 = 1000 nM T99089 CA9I0J 54580729 EC50 = 3700 nM T99089 CCJ4O1 54580890 IC50 = 3 nM T99089 C95MIN 54580891 IC50 = 4 nM T99089 CEL5N4 54580892 IC50 = 4 nM T99089 C9GWT2 54581065 IC50 = 660 nM T99089 CNQ0K4 54581121 IC50 = 410 nM T99089 C3S5AM 54581683 IC50 > 1000 nM T99089 CT8XP5 54581685 IC50 > 1000 nM T99089 C4X6DP 54581730 EC50 = 10000 nM T99089 C2KHN1 54581731 EC50 = 2900 nM T99089 CUDL04 54581778 IC50 = 37 nM T99089 CMZH76 54581779 IC50 = 3 nM T99089 CGL63B 54581944 IC50 = 5 nM T99089 C8MG6Q 54581945 IC50 = 670 nM T99089 CWQ62A 54582154 IC50 = 37.9 nM T99089 C7E8XC 54582155 IC50 = 8.1 nM T99089 CYJ3V4 54582156 IC50 = 10.7 nM T99089 C1V9TZ 54582157 IC50 = 350 nM T99089 CS87QB 54582674 IC50 = 647 nM T99089 CKV3C4 54582675 IC50 = 861 nM T99089 CS0PL6 54582676 IC50 = 0.66 nM T99089 CO87VE 54582742 IC50 = 8 nM T99089 CL7P3T 54582868 IC50 = 180 nM T99089 CAWE03 54582869 IC50 = 6 nM T99089 CBTW13 54583042 IC50 = 130 nM T99089 CO6B0E 54583043 IC50 = 7.9 nM T99089 CZRH05 54583044 IC50 = 2400 nM T99089 C6HCS1 54583107 IC50 = 970 nM T99089 CD4I8V 54583108 IC50 = 920 nM T99089 CDJ6G8 54583634 IC50 = 468 nM T99089 C4ZR2K 54583635 IC50 > 1000 nM T99089 C8ZRQ6 54583636 IC50 = 8 nM T99089 C2LUN7 54583637 IC50 = 0.57 nM T99089 CYU57L 54583878 IC50 = 799 nM T99089 C6K2HE 54584047 IC50 > 10000 nM T99089 CH9XG2 54584103 IC50 = 8 nM T99089 CV3E2I 54584104 IC50 = 600 nM T99089 CASX62 54584105 IC50 = 140 nM T99089 CSTH09 54584106 IC50 = 2000 nM T99089 C9ZC3U 54584611 IC50 > 1000 nM T99089 CK2Q9W 54584612 IC50 = 3.8 nM T99089 CD4B5P 54584613 IC50 = 3.2 nM T99089 CP7U4T 54584640 EC50 = 1000 nM T99089 CKFC13 54584711 IC50 = 3 nM T99089 CU8NQ4 54584712 IC50 = 21 nM T99089 C1O4MD 54584830 IC50 = 7 nM T99089 CD73TV 54584831 IC50 = 10 nM T99089 CE5B2W 54584832 IC50 = 4 nM T99089 C1XJW8 54584998 IC50 > 10000 nM T99089 CJ58MO 54584999 IC50 > 10000 nM T99089 C92ZHV 54585000 IC50 > 10000 nM T99089 C6Q8OC 54585001 IC50 = 110 nM T99089 C87OYZ 54585557 IC50 = 1540 nM T99089 C3BGY8 54585558 IC50 = 72.5 nM T99089 C0OY2N 54585559 IC50 = 4.6 nM T99089 CBUK26 54585560 IC50 = 1.25 nM T99089 C1D2OF 54585666 IC50 = 3 nM T99089 CLA1K6 54585957 IC50 > 10000 nM T99089 C3PGE2 54585958 IC50 = 25.7 nM T99089 CV7HJ8 54585959 IC50 = 2000 nM T99089 C2J4AW 54586018 IC50 = 450 nM T99089 CE18QV 54586536 IC50 = 23 nM T99089 C9LYS4 54586537 IC50 = 788 nM T99089 CZ9VQ3 54586538 IC50 = 3.7 nM T99089 CU0WR1 54586539 IC50 = 607 nM T99089 C5ITJ1 54586540 IC50 = 4.9 nM T99089 C7QWJ6 54586541 IC50 = 5 nM T99089 CFE96Y 54586652 IC50 = 3 nM T99089 CKI74Z 54586653 IC50 = 3 nM T99089 CJI6G8 54586767 IC50 = 5 nM T99089 CM31XW 54586768 IC50 = 5 nM T99089 CA4WF9 54586933 IC50 = 83 nM T99089 C0P7RF 54587401 IC50 = 13 nM T99089 CTB8J1 54587402 IC50 = 3 nM T99089 C6JVP8 54587568 IC50 > 1000 nM T99089 CQK04T 54587569 IC50 = 55 nM T99089 CRB13M 54587570 IC50 = 328 nM T99089 CS21RZ 54587660 IC50 = 7 nM T99089 CNB28I 54675261 IC50 = 32 nM T99089 CU9NY2 54675336 IC50 = 1.3 nM T99089 C6SW5P 54675374 IC50 = 0.2 nM T99089 CO6EN5 54675413 IC50 = 10 nM T99089 C6KE7Z 54675418 IC50 = 40 nM T99089 CLZ53I 54675419 IC50 = 6.3 nM T99089 C9SXQ0 54675442 IC50 = 8 nM T99089 C10VXC 54675444 IC50 = 79 nM T99089 CG35NE 54675446 IC50 = 16 nM T99089 CV6X5K 54675470 IC50 = 32 nM T99089 C4OZC7 54675473 IC50 = 1.3 nM T99089 C3YZ9F 54675501 IC50 = 0.6 nM T99089 C9YKJ7 54764764 IC50 = 8 nM T99089 CKV76W 54764765 IC50 = 10 nM T99089 CYFP20 54764766 IC50 = 6 nM T99089 CETW26 54764767 IC50 = 17 nM T99089 CEJR67 54764768 IC50 = 8 nM T99089 CY0TN4 56658293 IC50 = 2600 nM T99089 C6BE9H 56658294 IC50 = 530 nM T99089 CCY5N4 56658295 IC50 = 38 nM T99089 CP1W9R 56658296 IC50 = 18 nM T99089 CU36FV 56658297 IC50 = 29 nM T99089 C04BHC 56658298 IC50 = 38 nM T99089 CN8XD6 56658305 IC50 = 36 nM T99089 CLE4Y5 56658307 IC50 = 173 nM T99089 C4MJ5O 56658311 IC50 = 12 nM T99089 C7NP3M 56658312 IC50 = 1.8 nM T99089 CN4J9K 56658587 IC50 = 82 nM T99089 CH7Q4P 56659673 EC50 = 10 nM T99089 CN4U5R 56659674 EC50 = 8 nM T99089 C7I9AJ 56659836 EC50 = 7 nM T99089 CP2KY0 56661794 IC50 = 110 nM T99089 CN01KB 56661795 IC50 = 17 nM T99089 CJTU92 56661796 IC50 = 18 nM T99089 CBI7G3 56661797 IC50 = 19 nM T99089 CX62TD 56661798 IC50 = 200 nM T99089 CXE20W 56661799 IC50 = 400 nM T99089 CZ5XD1 56661804 IC50 = 80 nM T99089 C5XU3W 56661805 IC50 = 59 nM T99089 C6N0EJ 56661815 IC50 = 5.3 nM T99089 C91EDC 56661816 IC50 = 16 nM T99089 CG01XH 56662039 IC50 = 118 nM T99089 CFG9E7 56662196 IC50 = 113 nM T99089 C6RL1P 56663136 EC50 = 24 nM T99089 CBR9N7 56663302 IC50 = 9 nM T99089 CU0AC8 56663303 EC50 = 580 nM T99089 C2YO4N 56665241 IC50 = 61 nM T99089 C1DJ0Y 56665242 IC50 = 76 nM T99089 CE13AF 56665248 IC50 = 113 nM T99089 CJ85KT 56665256 IC50 = 4.2 nM T99089 C6VLY7 56665257 IC50 = 6.9 nM T99089 C4FD9N 56665258 IC50 = 0.5 nM T99089 C4RH8B 56665517 IC50 = 696 nM T99089 CKO56E 56668698 IC50 = 62 nM T99089 CJS5R1 56668699 IC50 = 100 nM T99089 CP0H1C 56668709 IC50 = 320 nM T99089 C7VMK6 56668710 IC50 = 0.2 nM T99089 C3C5MB 56668951 IC50 = 179 nM T99089 CH7G4I 56670002 IC50 = 1358 nM T99089 CQ1RX6 56670003 EC50 = 10 nM T99089 C8JY6A 56670156 EC50 = 52 nM T99089 CHFG31 56672169 IC50 = 150 nM T99089 CY8P0Z 56672170 IC50 = 29 nM T99089 CO65KN 56672171 IC50 = 120 nM T99089 CH37GX 56672177 IC50 = 96 nM T99089 C3BTJ1 56672436 IC50 = 290 nM T99089 CZXV87 56673516 EC50 = 11 nM T99089 C7YKI3 56673668 IC50 = 12 nM T99089 CC7T2A 56674921 IC50 = 190 nM T99089 CNF2C9 56675551 IC50 = 8.3 nM T99089 CA4RH3 56675552 IC50 = 170 nM T99089 CFU28L 56675553 IC50 = 25 nM T99089 C2JA0L 56675554 IC50 = 4.5 nM T99089 CGKN93 56675555 IC50 = 190 nM T99089 CRL0J4 56675556 IC50 = 40 nM T99089 CCAN48 56675557 IC50 = 140 nM T99089 CI17LQ 56675558 IC50 = 99 nM T99089 C31OWJ 56675570 IC50 = 46 nM T99089 C4CVI6 56675571 IC50 = 0.7 nM T99089 C4IR8B 56675821 IC50 = 1850 nM T99089 CO0U8T 56675936 IC50 = 229 nM T99089 CWB68U 56676987 IC50 = 5 nM T99089 CQK28C 56678886 IC50 = 110 nM T99089 C4ZX6A 56678887 IC50 = 13 nM T99089 C4FK3H 56678889 IC50 = 86 nM T99089 CJ47GL 56678899 IC50 = 1 nM T99089 CZ48XY 56679129 IC50 = 1664 nM T99089 C9NC2S 56680317 EC50 = 99 nM T99089 C8X0SE 56680318 IC50 = 1970 nM T99089 CM2H0R 56682202 IC50 = 1.4 nM T99089 C8SXR2 56682203 IC50 = 19 nM T99089 C64BDP 56682204 IC50 = 63 nM T99089 C5IQR3 56682205 IC50 = 33 nM T99089 CT1J5E 56682215 IC50 = 3.5 nM T99089 CQIS53 56682425 IC50 = 333 nM T99089 CH89ZU 56682426 IC50 = 10000 nM T99089 C19PCK 56683489 EC50 = 21 nM T99089 CV6GM9 56695913 IC50 = 1840 nM T99089 C1L5QU 56834881 IC50 = 58 nM T99089 CGEV72 56834882 IC50 = 2 nM T99089 C87YOZ 56929808 EC50 = 230 nM T99089 CGQ94I 56950740 IC50 > 100000 nM T99089 CN1XL0 56950741 IC50 > 100000 nM T99089 C3ER0V 56950742 IC50 = 64000 nM T99089 CEZ14X 56950743 IC50 > 100000 nM T99089 CTL49B 56950878 IC50 > 100000 nM T99089 CM5HO1 56950881 IC50 = 900 nM T99089 C9CLJ0 56950882 IC50 = 800 nM T99089 CG0VC7 56950883 IC50 = 860 nM T99089 CE1GO5 56950884 IC50 = 1400 nM T99089 CLQ4Z9 56950885 IC50 = 890 nM T99089 C40BPN 56951005 IC50 = 1700 nM T99089 CL9XP2 56951006 IC50 = 1500 nM T99089 CKV5O2 56951007 IC50 = 2500 nM T99089 C97QIR 56951008 IC50 = 2700 nM T99089 C61LYC 56951317 IC50 = 0.6 nM T99089 CB5V2D 56953628 IC50 = 101 nM T99089 C1A9IE 56953629 IC50 = 336 nM T99089 C48UTY 56953737 IC50 > 15000 nM T99089 CSPK46 56953738 IC50 = 355 nM T99089 C1ITV4 56953739 IC50 = 134 nM T99089 CO38GU 56953869 IC50 = 956 nM T99089 CS12TI 56953870 IC50 = 1134 nM T99089 CA2K6G 56953871 IC50 > 15000 nM T99089 CGBF17 56953872 IC50 = 649 nM T99089 C1ZQG0 56953873 IC50 = 324 nM T99089 CB83NX 56953992 IC50 = 645 nM T99089 CN7P1B 56953993 IC50 = 339 nM T99089 CI47JS 56953994 IC50 = 174 nM T99089 CIQJ93 56953995 IC50 = 308 nM T99089 C8DVS5 56953996 IC50 = 276 nM T99089 CL6W0K 56954119 IC50 = 109 nM T99089 CC31UP 56954120 IC50 = 183 nM T99089 C3BW5T 56954121 IC50 = 142 nM T99089 CKIC60 56954122 IC50 = 469 nM T99089 CN2L0O 56954123 IC50 = 84 nM T99089 CNH3A5 56954221 IC50 = 505 nM T99089 CE4YV5 56954222 IC50 = 681 nM T99089 CT95JA 56954223 IC50 > 1667 nM T99089 C73ZPH 56954224 IC50 = 21 nM T99089 C2ONU1 56954225 IC50 = 62 nM T99089 CL1IA3 56954309 IC50 = 1131 nM T99089 CNQ2G0 56955962 IC50 = 7 nM T99089 C7SJC2 56956247 IC50 = 3.02 nM T99089 C1FY0P 56965341 IC50 = 1 nM T99089 C01OBF 57342892 IC50 = 3400 nM T99089 CIWA26 57343054 IC50 = 9.5 nM T99089 CEOI16 57343055 IC50 = 0.1096 nM T99089 C4G7QD 57343225 IC50 = 0.18 nM T99089 C5DXS3 57343766 IC50 = 17 nM T99089 C32MLB 57343972 IC50 = 19 nM T99089 C8Q9ML 57344791 IC50 = 45 nM T99089 C89XBT 57344794 IC50 = 1 nM T99089 CT6H9M 57344795 IC50 = 9 nM T99089 C2WFQ3 57344993 IC50 = 18 nM T99089 CH71KO 57345095 IC50 = 41 nM T99089 C5YB9H 57345097 IC50 = 62 nM T99089 C3FY9A 57345328 IC50 = 1 nM T99089 CW9X3F 57386061 IC50 = 43 nM T99089 C8FS6P 57390778 IC50 = 15400 nM T99089 C13LDJ 57390779 IC50 = 2450 nM T99089 C3F0BW 57390780 IC50 = 38 nM T99089 CHY5D4 57390781 IC50 = 3 nM T99089 CC6ZD0 57390813 IC50 = 4 nM T99089 CB7KU9 57390814 IC50 = 1600 nM T99089 C82VXN 57391632 IC50 = 1780 nM T99089 CHI6C9 57392569 IC50 = 660 nM T99089 C4TXW2 57392593 IC50 = 3 nM T99089 CM8CB4 57392634 IC50 = 1210 nM T99089 CCP74G 57392635 IC50 = 212 nM T99089 CX2A5Y 57392636 IC50 = 1330 nM T99089 C7QGI8 57393255 IC50 = 290 nM T99089 CO0C5I 57394104 IC50 = 25000 nM T99089 CKVG97 57394105 IC50 = 26 nM T99089 CD2P1K 57394289 IC50 = 70 nM T99089 CDBV60 57394290 IC50 = 1 nM T99089 C1DAU4 57394291 IC50 = 390 nM T99089 CA75YZ 57394913 IC50 = 33.9 nM T99089 C8ZTY5 57394914 IC50 = 45.7 nM T99089 C0IJ9K 57394998 IC50 = 349 nM T99089 CKDR51 57395014 IC50 = 6.3 nM T99089 C13PQB 57395380 IC50 = 33 nM T99089 CO4WY9 57396045 IC50 = 180 nM T99089 C7EOQ2 57396104 IC50 = 67 nM T99089 CB1C3G 57396105 IC50 = 112 nM T99089 CE1VH5 57396728 IC50 = 1680 nM T99089 CO4QP1 57397207 IC50 = 2 nM T99089 CT4MN6 57397844 IC50 = 5300 nM T99089 C4J6UZ 57397845 IC50 = 45 nM T99089 C2JWM3 57397846 IC50 = 640 nM T99089 C8EM4N 57397875 IC50 = 28 nM T99089 CB47HC 57397876 IC50 = 40 nM T99089 CAN16F 57397919 IC50 = 14500 nM T99089 CZ1F9G 57397920 IC50 = 724 nM T99089 CT7D3Y 57398497 IC50 = 117 nM T99089 CN28HT 57398498 IC50 = 35 nM T99089 CM0C2E 57398516 IC50 = 35 nM T99089 C0BGR6 57399335 IC50 = 3 nM T99089 CS10GU 57399339 IC50 = 8600 nM T99089 CC04QG 57399505 IC50 = 2200 nM T99089 CVX1I4 57399506 IC50 = 600 nM T99089 C7DJ9Q 57399527 IC50 = 17 nM T99089 CPS08J 57399528 IC50 = 5 nM T99089 CVKR29 57399561 IC50 = 1540 nM T99089 C25ULW 57399562 IC50 = 5 nM T99089 CP0AL9 57399563 IC50 = 4 nM T99089 C1G6VF 57400171 IC50 = 18 nM T99089 CU4E6C 57400186 IC50 = 297 nM T99089 C7TAI9 57400292 IC50 = 1230 nM T99089 CJ7Y2K 57400603 IC50 = 2.2 nM T99089 CO63XJ 57401264 IC50 = 1300 nM T99089 C7BSY8 57401314 IC50 = 507 nM T99089 C3QEI9 57401315 IC50 = 275 nM T99089 C1IJV5 57401316 IC50 = 50 nM T99089 COZ7Q8 57401317 IC50 = 1120 nM T99089 C5UOF8 57401958 IC50 = 296 nM T99089 C0C6PE 57401959 IC50 = 293 nM T99089 CNVO29 57402060 IC50 = 3900 nM T99089 CX5O1I 57402078 IC50 = 1370 nM T99089 C6N8AU 57402861 IC50 = 1300 nM T99089 CL7MW8 57403007 IC50 = 150 nM T99089 CQH79M 57403036 IC50 = 4730 nM T99089 CA4L2E 57403037 IC50 = 14 nM T99089 CRJ9Q6 57403038 IC50 = 1 nM T99089 C2GYT1 57403706 IC50 > 10000 nM T99089 CB45FY 57403707 IC50 = 3470 nM T99089 C3R0XQ 57403708 IC50 = 3770 nM T99089 COQ75N 57403736 IC50 = 19 nM T99089 CA47JG 57433668 IC50 = 23 nM T99089 CE59QS 57505507 IC50 > 1000 nM T99089 C8P6RD 57505528 IC50 = 290 nM T99089 C4T7PW 57523998 IC50 = 31 nM T99089 C1Q7LS 57523999 IC50 = 195 nM T99089 CPS79I 57524088 IC50 = 54 nM T99089 C0CJ8Z 57524184 IC50 = 42 nM T99089 C8ICV2 57524400 IC50 = 58 nM T99089 CL72NQ 57524403 IC50 = 13 nM T99089 CAU0K1 57524478 IC50 = 53 nM T99089 C5FYG0 57568454 IC50 = 9 nM T99089 CN41VS 57568471 IC50 = 0.4 nM T99089 C5W4AZ 57568472 IC50 = 20 nM T99089 CE34TF 57568477 IC50 = 4 nM T99089 C6WMQ8 57568487 EC50 = 100 nM T99089 CW9L6C 57568544 IC50 = 1 nM T99089 CV1UP2 57568562 EC50 = 100 nM T99089 CK3NU1 57568594 IC50 < 0.4 nM T99089 CSA80G 57568606 IC50 = 10 nM T99089 CMR7A9 57568636 IC50 = 4 nM T99089 C6L9JH 57568638 EC50 = 400 nM T99089 C9AS4Q 57568659 IC50 < 0.4 nM T99089 CRF8M0 57708566 IC50 = 650 nM T99089 C4CJG6 57856282 IC50 = 6.5 nM T99089 CO1SN5 57989641 IC50 = 0.3 nM T99089 CJSR42 57989722 IC50 = 7 nM T99089 C61YOS 57989790 IC50 = 51 nM T99089 CHS76K 57989798 IC50 = 536 nM T99089 C9TN8I 57989818 IC50 = 28 nM T99089 C0FW7J 57989820 IC50 = 39.81 nM T99089 CR5IO7 57989894 IC50 = 1 nM T99089 CY5AF4 57989971 IC50 = 13 nM T99089 C1OV8I 57990029 IC50 = 10.96 nM T99089 CUPG23 57990033 IC50 = 28 nM T99089 C6BPR2 58985201 IC50 > 30000 nM T99089 CXT56U 59454465 IC50 = 170 nM T99089 CZ24KM 59454479 IC50 = 12 nM T99089 C5GV2P 59454483 IC50 = 13 nM T99089 C7N3LA 59454484 IC50 = 25 nM T99089 CCH48T 59454492 IC50 = 290 nM T99089 C8DT3V 59454506 IC50 = 18 nM T99089 C2BGR6 59506918 IC50 = 91 nM T99089 C0KZ6L 59507002 IC50 = 150 nM T99089 C6EJ9G 59507062 IC50 = 51 nM T99089 CHQK85 59507068 IC50 = 73 nM T99089 C8W5HT 59548263 IC50 > 1000 nM T99089 CVF1B2 59548283 IC50 > 1000 nM T99089 CC8UV3 59548383 IC50 > 1000 nM T99089 CD4ET2 59548402 IC50 > 1000 nM T99089 CES59T 59548403 IC50 > 1000 nM T99089 CBT21W 59548454 IC50 > 1000 nM T99089 CX8C2U 59548480 IC50 > 1000 nM T99089 CXJ63M 59603829 IC50 = 1500 nM T99089 CQEU96 59603842 IC50 = 19 nM T99089 CLH49Z 59790029 IC50 = 3 nM T99089 CW2GE7 59790182 EC50 = 100 nM T99089 C67DXJ 59823451 IC50 = 21.4 nM T99089 CN45KF 59823454 IC50 = 30.9 nM T99089 CZ2N7J 59823457 IC50 > 10000 nM T99089 CL4M6J 59823458 IC50 = 16.6 nM T99089 C8T6GZ 59823460 IC50 = 13.8 nM T99089 C27JOC 59823461 IC50 = 20.9 nM T99089 CGT41K 59823462 IC50 = 25.1 nM T99089 C5SC3K 59823463 IC50 = 19.5 nM T99089 C0K7JN 59823464 IC50 = 692 nM T99089 CNH9C6 59823465 IC50 = 9.6 nM T99089 C9QRX3 60098131 IC50 = 90 nM T99089 C9W0PE 60150671 IC50 = 570 nM T99089 C9NAL6 60152613 IC50 = 0.4 nM T99089 C5KD3Z 60154714 IC50 > 1000 nM T99089 CN0D8O 60154913 IC50 = 120 nM T99089 C9E6ZO 60154914 IC50 = 190 nM T99089 CS0L4D 60154996 IC50 > 1000 nM T99089 C59MPL 60154998 IC50 = 1600 nM T99089 CCO8H2 60154999 IC50 = 720 nM T99089 C1Z8VW 60155000 IC50 = 3600 nM T99089 C40TDP 60155001 IC50 = 520 nM T99089 C1UI3P 60155086 IC50 > 1000 nM T99089 C0DM1I 60165270 IC50 = 12 nM T99089 C46RPN 60196912 IC50 = 19 nM T99089 C52PMH 60196913 IC50 = 62 nM T99089 CTB23Y 60196914 IC50 = 2 nM T99089 C2Y9QK 60196916 IC50 = 8 nM T99089 CL90JM 60196917 IC50 = 814 nM T99089 C7FL4M 60197009 IC50 = 733 nM T99089 CD9ST6 60197011 IC50 = 18 nM T99089 C0Y2GI 60197014 IC50 = 17 nM T99089 C46JDT 60197113 IC50 = 11 nM T99089 CU69TF 60197114 IC50 = 100 nM T99089 CVB04X 60197118 IC50 = 44 nM T99089 C8IYB5 60197208 IC50 = 33 nM T99089 C8QY3Z 60197213 IC50 = 0.2 nM T99089 CF72YM 60197214 IC50 = 0.3 nM T99089 C5AUZ3 60197314 IC50 = 0.2 nM T99089 C8X4BC 60197315 IC50 = 0.2 nM T99089 CJBW03 60197316 IC50 = 0.3 nM T99089 C37IKA 60197416 IC50 = 3 nM T99089 CX2N4J 60197515 IC50 = 851 nM T99089 CP2YO9 60197609 IC50 = 603 nM T99089 CO32KC 60197610 IC50 = 110 nM T99089 CU93PB 66554192 IC50 = 300 nM T99089 CZ7Y1D 66563698 IC50 = 180 nM T99089 CCX0O1 66868153 IC50 = 239 nM T99089 C5TKV7 67053220 IC50 = 13 nM T99089 CU5IJ8 67053231 IC50 = 13 nM T99089 C34TLO 67155626 IC50 = 8.2 nM T99089 CV63UL 67240318 IC50 > 10000 nM T99089 CZJS42 67970606 IC50 = 7 nM T99089 CI9XT5 67970652 IC50 = 67 nM T99089 CGY3O4 67970808 IC50 = 8.2 nM T99089 C09NPT 67970942 IC50 = 149 nM T99089 C0V1YT 67971007 IC50 = 131 nM T99089 CTN06A 67971055 IC50 = 83 nM T99089 C2KVA0 67971197 IC50 = 19 nM T99089 C1ACK8 67971360 IC50 = 11 nM T99089 CWX29O 67991931 IC50 = 16 nM T99089 CX08WF 67995742 IC50 = 63 nM T99089 CH86NY 67995748 IC50 = 40 nM T99089 CE1C9K 67995854 IC50 = 50 nM T99089 C76ZXO 67995947 IC50 = 13 nM T99089 CHI27U 67995956 IC50 = 1 nM T99089 CQM36K 67996004 IC50 = 5 nM T99089 C1CWR6 67996103 IC50 = 79 nM T99089 C4SY7A 67996169 IC50 = 0.5 nM T99089 CJ0M7V 67996291 IC50 = 1 nM T99089 C02XNI 67996483 IC50 = 6 nM T99089 CQXI95 67996588 IC50 = 4 nM T99089 CW17YX 68281294 IC50 > 5000 nM T99089 CU57RD 68304261 IC50 = 250 nM T99089 CD9YL6 68304991 IC50 = 20 nM T99089 C24NDT 68305023 IC50 = 200 nM T99089 CT6D9Q 68305115 IC50 = 13 nM T99089 C0CEX5 68305269 IC50 = 2000 nM T99089 CYAS06 68305303 IC50 = 500 nM T99089 C3JE5H 68356029 IC50 = 371 nM T99089 CGM78B 68472574 IC50 = 2 nM T99089 CB8O4N 68475743 IC50 = 9.5 nM T99089 C5QZW4 68486699 IC50 = 36 nM T99089 CY0DU7 68489225 IC50 = 150 nM T99089 C68QHU 68490094 IC50 = 40 nM T99089 C4XJ6F 68513796 IC50 = 254 nM T99089 CAIO65 68796885 IC50 = 10 nM T99089 C5DGR9 69036886 IC50 = 2035 nM T99089 C4BT3M 69037249 IC50 = 1.2 nM T99089 C07ETL 69934912 IC50 = 6300 nM T99089 CL56IP 70648329 IC50 = 4 nM T99089 C90UOE 70648331 IC50 = 6 nM T99089 CM8VW3 70648666 IC50 = 6 nM T99089 C0FW2K 70648683 IC50 = 0.5 nM T99089 CE61CB 70648685 IC50 = 1 nM T99089 CO9VX3 70649090 IC50 = 8 nM T99089 C1WF5Y 70649102 IC50 = 32 nM T99089 CX1FS0 70649109 IC50 = 1 nM T99089 CQE6V9 70649110 IC50 = 1 nM T99089 CI7L1V 70649115 IC50 = 4 nM T99089 CD3FH7 70649129 IC50 = 6 nM T99089 C0L3KI 70649136 IC50 = 1 nM T99089 CQJ04E 70649137 IC50 = 1000 nM T99089 CRPZ67 70649546 IC50 = 0.6 nM T99089 CIP0R1 70681402 IC50 = 140 nM T99089 CR6QD9 70681403 IC50 > 10000 nM T99089 CU2R4E 70681940 IC50 = 7480 nM T99089 CCR80K 70683505 IC50 > 10000 nM T99089 CD7P4Z 70683506 IC50 > 10000 nM T99089 C6VYT3 70683507 IC50 = 10 nM T99089 C7WJV3 70683520 IC50 = 6 nM T99089 C4H1YN 70683521 IC50 = 0.5 nM T99089 C73WHU 70683665 IC50 = 407 nM T99089 C9THU7 70683668 IC50 = 80 nM T99089 C3ZY9V 70685605 IC50 = 128 nM T99089 CFMJ68 70685606 IC50 = 9 nM T99089 CMY8U3 70687757 IC50 = 72 nM T99089 CIL45P 70687767 IC50 = 15 nM T99089 C63NKC 70687931 IC50 > 10000 nM T99089 C94LEG 70688667 IC50 = 2000 nM T99089 CK6YS5 70689807 IC50 = 239.88 nM T99089 CAI8P9 70691945 IC50 = 338.84 nM T99089 CI6X1V 70691959 IC50 = 0.4 nM T99089 C9DB2A 70694163 IC50 > 10000 nM T99089 CF0L1C 70696119 IC50 = 3606 nM T99089 CT0WC5 70696120 IC50 = 71 nM T99089 CN6MQ5 70696121 IC50 = 13 nM T99089 CN6WH1 70696122 IC50 = 8.7 nM T99089 C7U9QP 70696131 IC50 = 0.5 nM T99089 CD7E8J 70702306 IC50 = 192 nM T99089 CO41NU 71449525 IC50 = 80 nM T99089 C1CQ6R 71450431 IC50 = 23 nM T99089 CAZ3X8 71451311 IC50 = 3.5 nM T99089 CJ1QX0 71451319 IC50 = 52 nM T99089 CEBO91 71452977 IC50 > 10000 nM T99089 CF83BP 71453141 IC50 = 1.9 nM T99089 CR84JX 71453419 IC50 > 1000 nM T99089 CC0B7J 71456634 IC50 = 39 nM T99089 CZ0JA6 71456644 IC50 = 1.3 nM T99089 CJ95FM 71456645 IC50 = 1.2 nM T99089 C4JN5B 71456646 IC50 = 0.7 nM T99089 C7X4MD 71456750 IC50 = 810 nM T99089 CHC18F 71458487 IC50 = 6.8 nM T99089 CY1J6W 71458499 IC50 = 5.1 nM T99089 CHQZ25 71459584 IC50 > 10000 nM T99089 C5HF2X 71460335 IC50 = 1 nM T99089 C4V5GM 71460336 IC50 = 0.9 nM T99089 CVR7F1 71461211 IC50 = 22 nM T99089 CZ6M0W 71462036 IC50 = 3 nM T99089 C37IZM 71518995 IC50 > 10000 nM T99089 C68LCK 71518996 IC50 = 4170 nM T99089 CGF07H 71518997 IC50 = 7940 nM T99089 CTS9V7 71524844 IC50 = 580 nM T99089 C18WLF 71524885 IC50 > 10000 nM T99089 CMB61W 71524886 IC50 > 10000 nM T99089 C1UAL5 71524887 IC50 > 10000 nM T99089 C12CBZ 71524888 IC50 > 10000 nM T99089 C79KSW 71524889 IC50 > 10000 nM T99089 CV1O5J 71524932 IC50 > 10000 nM T99089 C38WUT 71524933 IC50 > 10000 nM T99089 C0BQK4 71524934 IC50 = 330 nM T99089 C5OV9C 71524935 IC50 = 9400 nM T99089 C1SU3J 71524936 IC50 > 10000 nM T99089 C0MEX7 71524978 IC50 = 14000 nM T99089 CQ1C4P 71524979 IC50 > 10000 nM T99089 C85MJU 71524980 IC50 > 10000 nM T99089 C2OS9F 71524981 IC50 > 10000 nM T99089 CZ8T5O 71524982 IC50 = 3600 nM T99089 CT90UG 71525021 IC50 = 9 nM T99089 C2BX7R 71525024 IC50 = 42 nM T99089 CU69TN 71525025 IC50 = 29 nM T99089 CBF84J 71525027 IC50 > 100000 nM T99089 CHQK51 71525066 IC50 > 100000 nM T99089 CT9CH6 71525067 IC50 > 10000 nM T99089 CP41CH 71525069 IC50 = 1100 nM T99089 CYL6J2 71525070 IC50 > 10000 nM T99089 CFW37Q 71525071 IC50 > 10000 nM T99089 CUX15V 71525104 IC50 = 190 nM T99089 CY6S9V 71570573 IC50 = 360 nM T99089 CK1MO3 71570722 IC50 = 3 nM T99089 CYVP02 71570866 IC50 = 36 nM T99089 CPGN04 71582940 IC50 = 28.84 nM T99089 C53GDJ 71582941 IC50 = 300 nM T99089 C27PFR 71582942 IC50 = 100 nM T99089 CWG78B 71583043 IC50 = 208.93 nM T99089 C4W1XT 71583044 IC50 = 67 nM T99089 C5IGH7 71583154 IC50 = 168 nM T99089 C6O4RB 71583157 IC50 = 45 nM T99089 CXWE43 71583159 IC50 = 45 nM T99089 C8YQ4F 71583160 IC50 = 25 nM T99089 C3F8MJ 71583269 IC50 = 257.04 nM T99089 CG17NA 71583271 IC50 = 230 nM T99089 C6DO5H 71583273 IC50 = 74 nM T99089 CQP5V0 71583274 IC50 = 4 nM T99089 C8THY0 71583275 IC50 = 5 nM T99089 C9IOY7 71583377 IC50 = 8 nM T99089 CWO26F 71583378 IC50 = 38.9 nM T99089 CUYC39 71583380 IC50 = 10 nM T99089 C9HQR0 71583494 IC50 = 25 nM T99089 CCJ37F 71583495 IC50 = 430 nM T99089 CLB5J6 71583602 IC50 = 20 nM T99089 C2PZ5G 71583603 IC50 = 573 nM T99089 CW20DX 71583604 IC50 = 25 nM T99089 CZ31PU 71583657 IC50 = 230 nM T99089 CN8ZD6 71584271 IC50 = 398.11 nM T99089 CNH8G5 71584401 IC50 = 263.03 nM T99089 C56ICO 71584402 IC50 = 131.83 nM T99089 CQ4ZV3 71584403 IC50 = 369 nM T99089 CBX50I 71584404 IC50 = 917 nM T99089 CEJ69H 71584405 IC50 = 601 nM T99089 C72PUL 71584406 IC50 = 2290.87 nM T99089 CEXG64 71584539 IC50 = 5370.32 nM T99089 C8KHE0 71584540 IC50 = 777 nM T99089 CFJ45Z 71584541 IC50 = 330 nM T99089 CI5VT4 71584542 IC50 = 350 nM T99089 C8IG3A 71584543 IC50 = 280 nM T99089 CKCO49 71584544 IC50 = 89 nM T99089 CGM5P4 71584661 IC50 = 52.48 nM T99089 CA0GI1 71584662 IC50 = 130 nM T99089 CY28UI 71627417 IC50 = 22 nM T99089 C0XEQ1 71682500 IC50 > 5000 nM T99089 CRK2G6 71718268 IC50 = 16 nM T99089 CU83YL 71730951 IC50 = 18 nM T99089 C1TD4L 71731206 IC50 = 7.9 nM T99089 C7F3ZM 71736390 IC50 = 8.4 nM T99089 C9EM5X 71736552 IC50 = 4.3 nM T99089 CKYO24 71736864 IC50 = 18 nM T99089 CA1JH2 71815073 IC50 = 190 nM T99089 C1E4RK 71818600 IC50 = 19 nM T99089 CX78NJ 71818601 IC50 = 18 nM T99089 C8WZ1R 71818732 IC50 = 14 nM T99089 C4B7ZW 71818733 IC50 = 9.5 nM T99089 C0QBF6 72375428 IC50 = 3.4 nM T99089 CL14JN 73330891 IC50 = 3.15 nM T99089 CXW8L5 73330892 IC50 = 2.78 nM T99089 CK9ST7 73330893 IC50 = 1.2 nM T99089 CINP24 73330894 IC50 = 19.1 nM T99089 CK3FN2 73331037 IC50 = 29.4 nM T99089 CX2I7B 73331038 IC50 = 1.03 nM T99089 CJC7V0 73331039 IC50 = 7.13 nM T99089 CMJY29 73331040 IC50 = 1.6 nM T99089 CB96JV 73331041 IC50 = 1.3 nM T99089 CKT5E7 73331182 IC50 = 2.17 nM T99089 CNO0C9 73331183 IC50 = 3.62 nM T99089 C7PI5W 73331184 IC50 = 1.5 nM T99089 C4CRH9 73331185 IC50 = 4.82 nM T99089 C0FYW2 73331186 IC50 = 8.07 nM T99089 C6XHO8 73331320 IC50 = 0.79 nM T99089 C6TA4H 73331323 IC50 = 2.51 nM T99089 CU60BO 73331324 IC50 = 2.71 nM T99089 CF3C1P 73331464 IC50 = 3.03 nM T99089 CEAF70 73425627 IC50 = 0.8 nM T99089 CD84TH 73425628 IC50 = 0.8 nM T99089 C2UGD3 73425629 IC50 = 0.1 nM T99089 C3QDX5 73425728 IC50 = 0.6 nM T99089 CC7GL1 73427048 IC50 = 70 nM T99089 CF2C5V 73427050 IC50 = 11 nM T99089 CJPU56 73427150 IC50 = 220 nM T99089 CX5K0Z 73427151 IC50 = 7 nM T99089 CQJ0R1 73427152 IC50 = 80 nM T99089 C1QFO2 73427153 IC50 = 7 nM T99089 CKI3Z2 73427155 IC50 = 7 nM T99089 C80SEC 73504974 IC50 = 187 nM T99089 CK1BY2 73504975 IC50 = 165 nM T99089 CE79YJ 73505176 IC50 = 1780 nM T99089 CC75WA 73505177 IC50 = 3260 nM T99089 C2LGB5 73505178 IC50 = 4060 nM T99089 CFG01S 73505179 IC50 = 942 nM T99089 C3KVB2 73505180 IC50 = 73 nM T99089 C0JF6O 75596779 IC50 = 157 nM T99089 C5BV3G 76310396 IC50 = 880 nM T99089 CX4H6I 86583042 IC50 = 8 nM T99089 CVR43W 86583044 IC50 > 1000 nM T99089 CA81UY 86583045 IC50 > 1000 nM T99089 CI2CG1 89670173 IC50 = 23 nM T99089 C1HW4B 89735655 IC50 = 1100 nM T99089 C7TJR3 89814000 IC50 = 27 nM T99089 C4WP7D 89827799 IC50 = 7.7 nM T99089 CZJ8N6 90116353 IC50 = 3.5 nM T99089 CB7R6C 90116945 IC50 = 4.2 nM T99089 CNR6C3 90120675 IC50 = 31 nM T99089 C6RZ7J 90408826 IC50 = 0.4 nM T99089 CW61DN 90488999 IC50 = 2.1 nM T99089 CY9FE6 90655275 IC50 = 551 nM T99089 C1CFP6 90655276 IC50 = 573 nM T99089 CI8XW3 90655277 IC50 = 110 nM T99089 CT28VM 90655278 IC50 = 240 nM T99089 C8N5TF 90655279 IC50 = 280 nM T99089 CPN1I6 90655280 IC50 = 670 nM T99089 CW1LJ4 90655281 IC50 = 410 nM T99089 CAC3D4 90655282 IC50 > 10000 nM T99089 CKO3Z1 90655283 IC50 = 290 nM T99089 C7S8KR 90655284 IC50 = 510 nM T99089 CY0T9O 90655285 IC50 = 340 nM T99089 CG9HX4 90655286 IC50 = 390 nM T99089 C7DT3G 90655287 IC50 = 230 nM T99089 C8RA1Y 90655288 IC50 = 37 nM T99089 C1B7TW 90655289 IC50 = 210 nM T99089 CVO26Z 90655290 IC50 = 300 nM T99089 CO5M8T 90655291 IC50 = 48 nM T99089 CXNB56 90655292 IC50 = 220 nM T99089 CW08SL 90655293 IC50 = 48 nM T99089 CC2P7K 90655294 IC50 = 360 nM T99089 CBX47C 90655295 IC50 = 290 nM T99089 CWD4O3 90655989 IC50 > 50000 nM T99089 CMH6T8 90664306 IC50 = 1.6 nM T99089 CND1X5 90670915 IC50 = 314 nM T99089 C92HCD 102531936 EC50 < 500 nM T99089 C4MBJ3 102531937 IC50 < 100 nM T99089 C4UTP7 102531938 IC50 < 100 nM T99089 CTGP06 117996541 IC50 = 416.87 nM T99089 CY3L2E 117996700 IC50 > 10000 nM T99089 CVP10Z 117996749 IC50 = 2900 nM T99089 CG7QL4 118705925 IC50 = 38.3 nM T99089 C4AHL2 118711367 IC50 > 10000 nM T99089 C5E6DW 118720154 IC50 = 12 nM T99089 C0XWT1 118720155 IC50 = 4.21 nM T99089 CKA6P4 118720156 IC50 = 13.5 nM T99089 C63KJT 118720157 IC50 = 10.8 nM T99089 C9UQA1 118720457 IC50 = 0.669 nM T99089 CRJ82K 118720458 IC50 = 2.56 nM T99089 CS45ZU 118720459 IC50 = 1.77 nM T99089 CQP9B3 118720460 IC50 = 7.44 nM T99089 C5OIW3 118720461 IC50 = 471 nM T99089 CWQC25 118720462 IC50 = 6430 nM T99089 C3KLI5 118723185 IC50 > 100000 nM T99089 CD1RU5 118725683 IC50 = 2470 nM T99089 C17SHY 118725687 IC50 = 40400 nM T99089 CZVH46 118725690 IC50 = 650 nM T99089 C6GQL2 118725758 IC50 = 531 nM T99089 C5QC8E 118730408 IC50 > 1000 nM T99089 C4TXF2 118730409 IC50 > 1000 nM T99089 CN2A9O 118730410 EC50 = 190 nM T99089 COF69K 118730411 IC50 = 8 nM T99089 CEJ1S6 118730412 IC50 = 66 nM T99089 CQ0T5Z 118730413 IC50 = 13 nM T99089 CF47CO 118730414 IC50 > 1000 nM T99089 CEJ67D 118730415 IC50 > 1000 nM T99089 C5SI6Q 118730416 IC50 > 1000 nM T99089 CR0H9D 118730417 IC50 > 1000 nM T99089 CGDW48 118730418 IC50 > 1000 nM T99089 C23KFD 118730419 IC50 > 1000 nM T99089 CJ9SA8 118730420 IC50 > 1000 nM T99089 C0HK5A 118730421 IC50 > 1000 nM T99089 C1Q0UN 118730422 IC50 > 1000 nM T99089 C1K0PE 118730423 IC50 > 1000 nM T99089 CQCX41 118737057 IC50 = 15 nM T99089 CESI90 118988423 IC50 = 54 nM T99089 C0UT7G 122177477 IC50 = 6.8 nM T99089 CSF49R 122177478 IC50 = 40 nM T99089 CDQ60H 122179517 IC50 = 149 nM T99089 CS07QW 122179518 IC50 = 177 nM T99089 C6HB9Q 122179519 IC50 = 68 nM T99089 CH6C3N 122179520 IC50 = 917 nM T99089 C4P2OM 122179521 IC50 = 593 nM T99089 CQ52KS 122179522 IC50 = 51 nM T99089 CBS2G4 122179523 IC50 = 48 nM T99089 CXN92S 122179524 IC50 = 4310 nM T99089 CQ48MD 122179525 IC50 = 533 nM T99089 CHC9Z8 122179526 IC50 = 17 nM T99089 CSFU53 122179527 IC50 = 122 nM T99089 CRH7W6 122179528 IC50 = 25 nM T99089 CKFP69 122179529 IC50 = 10 nM T99089 C9KF6J 122179530 IC50 = 16 nM T99089 CG3OM1 122179531 IC50 = 3 nM T99089 C29LPV 122179532 IC50 = 131 nM T99089 CO5TH2 122179533 IC50 = 107 nM T99089 CAPV50 122179534 IC50 = 21 nM T99089 CL4OW0 122179535 IC50 = 11 nM T99089 C08KEM 122179540 IC50 = 2500 nM T99089 CG0RP7 122179547 IC50 = 6200 nM T99089 C1A0SQ 122179548 IC50 = 5900 nM T99089 C5B6QT 122189918 IC50 = 668 nM T99089 COWC81 127025601 IC50 = 2.9 nM T99089 C1HGA4 127025889 IC50 = 2.1 nM T99089 CF61HD 127025890 IC50 = 74 nM T99089 CM74CE 127025891 IC50 = 34 nM T99089 CAPU43 127026035 IC50 > 30 nM T99089 CQVU25 127026051 IC50 = 17 nM T99089 CZVP92 127028061 IC50 = 67 nM T99089 CZ3G8X 127028062 IC50 = 854 nM T99089 C2KCN9 127028071 IC50 > 12500 nM T99089 CN32ML 127028362 IC50 = 2.9 nM T99089 C1K5UC 127028929 IC50 = 20 nM T99089 C6KM3T 127034964 IC50 = 2 nM T99089 CF5WH1 127039888 IC50 = 7820 nM T99089 CH09EC 127041357 IC50 > 12500 nM T99089 C0D7RE 127042274 IC50 > 12500 nM T99089 C6NZ1Q 127042619 IC50 > 12500 nM T99089 CS2AP8 127042622 IC50 = 2.7 nM T99089 CL40ZB 127042623 IC50 = 3.1 nM T99089 CJ45OF 127042624 IC50 = 45 nM T99089 C3NMP8 127042932 IC50 = 5010 nM T99089 CP9L4A 127042940 IC50 = 1.9 nM T99089 CJ1G3I 127045769 IC50 = 1 nM T99089 CKL75H 127045770 IC50 = 1 nM T99089 CN7Z1E 127045771 IC50 = 216 nM T99089 CHM08S 127045839 IC50 = 141 nM T99089 C8W9VK 127045991 IC50 = 177 nM T99089 C2S9ZM 127046079 IC50 = 57 nM T99089 CFP01I 127046080 IC50 = 44 nM T99089 C8LRC5 127046081 IC50 = 15 nM T99089 C1BLZ3 127046082 IC50 = 122 nM T99089 CGO7P6 127046232 IC50 = 420 nM T99089 C9P5OW 127046289 IC50 = 68 nM T99089 CM05VG 127046445 IC50 = 17 nM T99089 CJZ6X2 127046446 IC50 = 26 nM T99089 CNA7K2 127046457 IC50 = 13 nM T99089 CC2AP7 127046458 IC50 = 240 nM T99089 CJ8V6Q 127046459 IC50 = 453 nM T99089 CSX5M4 127046460 IC50 = 38 nM T99089 CN26AU 127046461 IC50 = 2031 nM T99089 CAG9K7 127046489 IC50 = 95 nM T99089 CA6WZ4 127046615 IC50 = 5 nM T99089 CR7V4J 127047050 IC50 = 3 nM T99089 C2UBH1 127047051 EC50 = 1510 nM T99089 C7U9GE 127047125 IC50 = 563 nM T99089 CKU72G 127047243 IC50 = 2 nM T99089 C7P9XY 127047244 IC50 = 26 nM T99089 CFBT16 127047245 IC50 = 356 nM T99089 CK5XG8 127047246 IC50 = 22 nM T99089 C6DP7Y 127047275 IC50 = 131 nM T99089 C3DVM9 127047276 IC50 = 1230 nM T99089 CXK40B 127047368 IC50 > 10000 nM T99089 CEND36 127047369 IC50 > 10000 nM T99089 C34NAH 127047506 IC50 = 785 nM T99089 C2GA5N 127047507 IC50 = 1512 nM T99089 C38WDB 127047508 IC50 = 3530 nM T99089 CLXZ13 127047509 IC50 = 1210 nM T99089 CHC2M7 127047632 IC50 = 110 nM T99089 C0U1FB 127047676 IC50 = 1000 nM T99089 C3YWV1 127047786 IC50 = 50 nM T99089 CLPC17 127047787 IC50 = 125 nM T99089 C81LVM 127047788 IC50 = 1030 nM T99089 C12AUN 127047893 IC50 = 111 nM T99089 CMBQ27 127047908 IC50 = 182 nM T99089 COTB30 127047909 IC50 = 434 nM T99089 CM81AR 127047922 IC50 = 4300 nM T99089 CRV7N4 127048021 IC50 = 27 nM T99089 C4JKZ1 127048022 EC50 = 8090 nM T99089 C67PQF 127048023 IC50 = 4 nM T99089 CC7IS1 127048327 IC50 = 1490 nM T99089 CK03IO 127048328 IC50 = 610 nM T99089 C2KYI6 127048329 IC50 = 230 nM T99089 C1JZ8I 127048676 IC50 = 720 nM T99089 CLN2V6 127048677 IC50 = 2540 nM T99089 CP6D8F 127048678 IC50 = 670 nM T99089 CBEM37 127049658 IC50 > 10000 nM T99089 CJG89B 127049660 IC50 = 840 nM T99089 C6OP7G 127049661 IC50 = 55 nM T99089 CP9T1K 127049662 IC50 = 420 nM T99089 CW0Y3A 127049663 IC50 = 60 nM T99089 CB2M4K 127049664 IC50 = 210 nM T99089 CSV6H4 127049665 IC50 = 1640 nM T99089 CT6W1K 127049960 IC50 > 10000 nM T99089 C1CFZ7 127049961 IC50 = 300 nM T99089 CGWP70 127049962 IC50 = 9870 nM T99089 C4KAX3 127049963 IC50 > 10000 nM T99089 CAQL02 127049964 IC50 > 10000 nM T99089 C0FU7Y 127049965 IC50 = 200 nM T99089 C0XS1L 127051137 IC50 = 1000 nM T99089 C0AJS1 127051166 IC50 > 10000 nM T99089 CQ1K5O 127051167 IC50 > 10000 nM T99089 CKC0Z6 127051168 IC50 > 10000 nM T99089 CA91BN 127051468 IC50 = 5920 nM T99089 CV3L6M 127052123 IC50 = 1200 nM T99089 CTV2I4 127052124 IC50 > 10000 nM T99089 CJ21BE 127052125 IC50 > 10000 nM T99089 CVB1C9 127052416 IC50 = 130 nM T99089 C74KCH 127052706 IC50 = 250 nM T99089 C0FM1R 130196825 IC50 = 8294 nM T99089 CM2J3B 131953483 IC50 > 1000 nM T99089 CBI35E 132275094 IC50 = 14 nM T99089 CU1H0W 132497402 IC50 = 77.2 nM T99089 CSZA35 134133678 IC50 = 10120 nM T99089 CXSB18 134133754 IC50 = 22010 nM T99089 CRH7A2 134135364 IC50 = 1760 nM T99089 C62GWK 134141404 IC50 = 2400 nM T99089 C4QT7E 134142822 IC50 > 50000 nM T99089 C7I5JQ 134144573 IC50 = 2560 nM T99089 CDMB08 134145603 IC50 > 50000 nM T99089 CVNG59 134145628 IC50 = 8930 nM T99089 CMY13K 134146982 IC50 = 24230 nM T99089 CUZ48A 134149722 IC50 = 680 nM T99089 CU4T3D 134149937 IC50 = 33490 nM T99089 CYL31R 134150731 IC50 = 280 nM T99089 C8OP5K 134151586 IC50 = 3270 nM T99089 CC3Y0N 134152150 IC50 = 1840 nM T99089 C9B6PV 134152705 IC50 = 370 nM T99089 C8WVZ0 134152967 IC50 = 2900 nM T99089 CPZ10X 134155617 IC50 = 17810 nM T99089 C29UML 134155621 IC50 = 1800 nM T99089 CMPS85 134155826 IC50 = 920 nM T99089 C2AN7T 134611886 IC50 > 100000 nM T99089 CX1FA8 135399664 IC50 < 2 nM T99089 CKY3I2 135401910 IC50 = 0.2 nM T99089 C2H0FA 135401911 IC50 < 2 nM T99089 C85QZP 135453073 IC50 = 18000 nM T99089 CHJU83 135466457 IC50 = 0.15 nM T99089 CQ7L2Y 135482542 IC50 = 29420 nM T99089 CMW1V4 135505774 IC50 = 16 nM T99089 C2GQW0 135508240 IC50 = 0.48 nM T99089 C8B5GZ 135513879 IC50 = 339 nM T99089 CEK31P 135566415 IC50 > 20000 nM T99089 C8P7BR 135688666 IC50 > 100000 nM T99089 CX4ZB3 135863110 IC50 > 10000 nM T99089 C30RIL 135895396 IC50 = 250 nM T99089 CC7J0Q 135923565 IC50 = 4900 nM T99089 CJL23B 135936239 IC50 = 130 nM T99089 C51AMW 135981332 IC50 = 720 nM T99089 CG9PJ7 135993841 IC50 = 655.2 nM T99089 CN47FL 136030704 IC50 = 35 nM T99089 CDYC36 136030724 IC50 = 16 nM T99089 CW7G2B 136042252 IC50 = 954 nM T99089 C5HUM3 136045809 IC50 = 18.4 nM T99089 CZU9M0 136073752 IC50 = 110 nM T99089 CG1R7B 136087060 IC50 > 10000 nM T99089 C8YZS6 136141580 IC50 = 47 nM T99089 C3COS8 136160805 IC50 = 0.5 nM T99089 CGKV52 136164074 IC50 = 1600 nM T99089 CZ7EX0 136183413 IC50 > 30000 nM T99089 CI6V9T 136192928 IC50 = 4 nM T99089 C4KSL5 136235605 IC50 = 8800 nM T99089 C4P5VI 137631729 IC50 > 10000 nM T99089 C4N0LW 137631825 IC50 > 1000 nM T99089 C7NFX9 137632089 IC50 = 24.1 nM T99089 C9OV8U 137632895 IC50 = 140 nM T99089 C4JIL5 137633313 IC50 = 46.1 nM T99089 C51IZU 137633597 IC50 = 25.1 nM T99089 CI1E8V 137634241 IC50 > 10000 nM T99089 CP8UG5 137634530 IC50 = 0.3 nM T99089 CN4BD6 137634880 IC50 = 21.4 nM T99089 C95VXH 137634988 IC50 = 39.1 nM T99089 C2FGN9 137635830 IC50 = 68.2 nM T99089 C8DTW2 137636634 IC50 = 135 nM T99089 C08MHJ 137636777 IC50 = 2.8 nM T99089 C0OWY3 137636794 IC50 > 10000 nM T99089 CV3A5G 137637973 IC50 = 60 nM T99089 COT76N 137638146 IC50 = 38.6 nM T99089 C3M5ET 137638260 IC50 = 8.4 nM T99089 C7TN8O 137639492 IC50 = 22.4 nM T99089 COBX17 137640041 IC50 = 441 nM T99089 CF5I3U 137640119 IC50 = 59.5 nM T99089 C0SJ2W 137640898 IC50 = 4.3 nM T99089 CA13KP 137642491 IC50 = 18.7 nM T99089 CDG2S9 137643098 IC50 = 152 nM T99089 CRI78Y 137643278 IC50 = 143 nM T99089 C9SOI8 137644117 IC50 > 2000 nM T99089 CHM1K2 137644157 IC50 = 88.6 nM T99089 C23ACF 137644903 IC50 > 2000 nM T99089 CQS67M 137644972 IC50 > 5000 nM T99089 CL8W4P 137647062 IC50 = 14.3 nM T99089 CIJK82 137647304 IC50 > 10000 nM T99089 C97LQG 137647372 IC50 = 169.2 nM T99089 C0KZ9Q 137647934 IC50 = 201 nM T99089 CGQ02E 137648059 IC50 = 10.5 nM T99089 CZ2B1S 137648159 IC50 = 30.8 nM T99089 CB7M8Z 137648383 IC50 = 21.6 nM T99089 CL9HT1 137648599 IC50 = 19.5 nM T99089 C8FV4X 137649404 IC50 = 35.8 nM T99089 CJMW91 137649638 IC50 > 1000 nM T99089 CNTC73 137649645 IC50 = 80.2 nM T99089 CF1H4X 137650051 IC50 > 10000 nM T99089 C1BUD8 137650370 IC50 = 145 nM T99089 CE7KF3 137650390 IC50 = 12.2 nM T99089 C3O6KY 137652367 IC50 = 29.1 nM T99089 CBVE69 137652761 IC50 = 388 nM T99089 CYMU46 137654572 IC50 = 178 nM T99089 CHSL51 137654792 IC50 = 43.1 nM T99089 CVCD38 137654923 IC50 = 18.3 nM T99089 CF8HI3 137655054 IC50 = 44.1 nM T99089 CF2PV0 137655959 IC50 = 901.8 nM T99089 C21RYV 137656620 IC50 = 237 nM T99089 CMPJ36 137656808 IC50 = 21.2 nM T99089 C6Y8BI 137656893 IC50 = 31.5 nM T99089 CHF87V 137657244 IC50 > 1000 nM T99089 CN7J2A 137657347 IC50 > 10000 nM T99089 CVQF35 137659532 IC50 = 251 nM T99089 C2VQL7 137660816 IC50 = 13.9 nM T99089 CZ4WT5 137661137 IC50 = 18.5 nM T99089 C1W3PN 137661841 IC50 > 1000 nM T99089 CA4V9R 137661906 IC50 = 260 nM T99089 C2JI6T 138393294 IC50 > 1000 nM T99089 C68OZS 138403232 IC50 = 420 nM T99089 CK90OA 138753620 IC50 = 272.3 nM T99089 COB9P2 141456067 IC50 = 3400 nM T99089 C6CN8H 142739455 IC50 = 316 nM T99089 C6VB3O 145925651 IC50 >= 5000 nM T99089 CB3Z1W 145949428 IC50 = 32 nM T99089 CT25FH 145950796 IC50 = 23.6 nM T99089 CHKS76 145952159 IC50 = 215.6 nM T99089 C1G0PH 145952494 IC50 = 407.2 nM T99089 C9WYS2 145954493 IC50 = 40.9 nM T99089 CF1T9Y 145954667 IC50 = 171.5 nM T99089 CX80ZF 145954847 IC50 = 85.2 nM T99089 CBR2Q7 145956253 IC50 = 476.3 nM T99089 C5VSC7 145956704 IC50 = 20 nM T99089 CZ3G0H 145959478 IC50 = 487.8 nM T99089 C7RQ8I 145960033 IC50 = 105.6 nM T99089 C7O0EG 145964682 EC50 = 240 nM T99089 CT49MR 145965412 IC50 = 6 nM T99089 C4NP2V 145965631 IC50 > 50000 nM T99089 C9H4TP 145966705 EC50 = 540 nM T99089 CR6O2S 145967668 IC50 = 5851 nM T99089 C49QZE 145967671 IC50 = 158 nM T99089 C0UZ6Q 145967831 IC50 = 1785 nM T99089 C2CHJ9 145967839 IC50 = 810 nM T99089 C5E8ZK 145968310 IC50 = 27 nM T99089 CTX9I2 145968517 IC50 = 69 nM T99089 C0Y1IT 145968532 IC50 = 973 nM T99089 CL0BO5 145968619 IC50 > 10000 nM T99089 CHAU61 145968737 IC50 = 21 nM T99089 CK1N7F 145968871 IC50 = 93 nM T99089 CBJ0F1 145968889 IC50 = 503 nM T99089 C0BG4F 145968971 IC50 = 442 nM T99089 CFC48X 145969905 IC50 = 791 nM T99089 C4D3BL 145970607 IC50 = 33 nM T99089 C8NK3O 145970839 IC50 = 17 nM T99089 CP6QH1 145971042 IC50 = 9866 nM T99089 C87WHG 145973554 IC50 = 0.3 nM T99089 CLN2D9 145973734 EC50 = 480 nM T99089 C76RQZ 145976309 IC50 = 0.9 nM T99089 CBR8K6 145976838 IC50 = 3900 nM T99089 C59VIT 145977243 IC50 > 50000 nM T99089 C93ZOX 145977611 IC50 = 5 nM T99089 CG9BL6 145979052 IC50 = 39300 nM T99089 C2I5WD 145979310 IC50 = 29.7 nM T99089 C0DOU5 145979395 IC50 = 510 nM T99089 CQ03XU 145980353 IC50 > 200000 nM T99089 C16ENO 145980866 IC50 = 223.87 nM T99089 CTC34W 145981191 IC50 = 21300 nM T99089 CI24XE 145981336 IC50 > 200000 nM T99089 CJPU41 145981957 IC50 = 1000 nM T99089 C6T4MU 145982183 IC50 = 19 nM T99089 CSWY46 145982727 IC50 = 73.9 nM T99089 CIYQ21 145982961 IC50 = 5.75 nM T99089 CBR08X 145983359 IC50 = 13 nM T99089 CE2X6V 145983518 IC50 = 44 nM T99089 C4QE7K 145983757 IC50 = 2600 nM T99089 CFRC51 145984297 IC50 = 73.8 nM T99089 CLV2K6 145984391 IC50 > 200000 nM T99089 C1DM4I 145984486 IC50 = 2900 nM T99089 COPW70 145984516 IC50 = 2700 nM T99089 C4ID8J 145984666 IC50 = 51 nM T99089 C06ECS 145984689 IC50 = 352 nM T99089 C05VIR 145984747 IC50 = 46 nM T99089 CGT8Z5 145984754 IC50 = 168 nM T99089 CW6ZJ2 145984860 IC50 = 87 nM T99089 CI1VH9 145985185 IC50 > 200000 nM T99089 CR91FS 145985335 IC50 = 24 nM T99089 CSQ34B 145985725 IC50 = 20.3 nM T99089 CQ5S2M 145985741 IC50 = 421 nM T99089 CL3HZ6 145986481 IC50 = 48900 nM T99089 C10TUA 145986573 IC50 = 280 nM T99089 CS78MW 145986924 IC50 = 156000 nM T99089 C1FE9Y 145987180 IC50 = 4.786 nM T99089 C96XWA 145987467 IC50 = 1.698 nM T99089 CK8S4V 145988419 IC50 = 48 nM T99089 CI7M2B 145988861 IC50 = 12.6 nM T99089 CNLH48 145988888 IC50 = 18700 nM T99089 CBC9Q6 145989837 IC50 = 61 nM T99089 CMQG17 145990430 IC50 = 1360 nM T99089 CB0AC5 145990447 IC50 = 5210 nM T99089 C2GWJ6 145990512 IC50 = 124000 nM T99089 C3WRL8 145990775 IC50 > 200000 nM T99089 CC1Z8Y 145991567 IC50 = 23100 nM T99089 CR76UY 145991825 IC50 = 35600 nM T99089 C6UNJ7 145992396 IC50 = 95900 nM T99089 CRT48W 145993502 IC50 = 5230 nM T99089 CF57DG 146020550 IC50 = 125.7 nM T99089 CCO93U 154634893 IC50 = 453 nM T99089 C5DMK6 154634900 IC50 > 1000 nM T99089 CVY7N6 154634909 IC50 = 795 nM T99089 C7YD9F 154634910 IC50 > 1000 nM T99089 CE4V9P 154634911 IC50 = 856 nM T99089 C9CQ3T 154634913 IC50 = 272 nM T99089 CEC1D3 154634916 IC50 > 1000 nM T99089 CGO62P 154634918 IC50 = 190 nM T99089 C41FIQ 154634920 IC50 = 39 nM T99089 C6XWC7 154634922 IC50 = 334 nM T99089 C2NKF8 155076930 IC50 = 13.4 nM T99089 CY1ZH2 155510358 IC50 = 158 nM T99089 CB0IE5 155511260 IC50 = 2600 nM T99089 C0O5DS 155511991 IC50 = 3.9 nM T99089 C73ZFN 155512053 IC50 = 390 nM T99089 CZ5S2M 155512875 IC50 = 3.5 nM T99089 C1LC2I 155513138 IC50 = 0.2 nM T99089 C2MD1Q 155513187 IC50 > 10000 nM T99089 C8DAU4 155513645 IC50 = 7.4 nM T99089 C60ASE 155514455 IC50 = 7 nM T99089 CI54TD 155514548 IC50 = 3740 nM T99089 C2BA1L 155514841 IC50 = 6320 nM T99089 CX2E0D 155514846 IC50 = 7410 nM T99089 CX8LF1 155515119 IC50 = 100 nM T99089 CX6SR0 155516442 IC50 = 940 nM T99089 C13KCF 155517164 IC50 = 83.1 nM T99089 C40CDF 155518050 IC50 = 9 nM T99089 CS31UH 155519078 IC50 = 5320 nM T99089 CMH01P 155519212 IC50 = 189 nM T99089 C3M6GZ 155519761 IC50 = 220 nM T99089 CEZ4O1 155520166 IC50 = 198 nM T99089 C2IC0U 155520258 IC50 = 320 nM T99089 CRNT47 155520316 IC50 = 87200 nM T99089 CU6Z5O 155520650 IC50 = 110 nM T99089 C8P6FS 155520920 IC50 > 300 nM T99089 CP4JL5 155521754 IC50 < 10000 nM T99089 CM3DB7 155523430 IC50 = 1290 nM T99089 CLB37N 155524340 IC50 = 919 nM T99089 CD2U5W 155524889 IC50 = 212 nM T99089 C6BAZ7 155525737 IC50 = 14 nM T99089 CYZ16N 155526190 IC50 > 1000 nM T99089 CZQ8D2 155526237 IC50 = 4170 nM T99089 C3QDI9 155526245 IC50 = 6.2 nM T99089 C46UIC 155526269 IC50 = 688 nM T99089 CH87DO 155527260 IC50 = 21 nM T99089 C6AGH4 155527315 IC50 > 1000 nM T99089 CH02ZE 155530305 IC50 = 45 nM T99089 CL0V4U 155530858 IC50 = 640 nM T99089 CLY07C 155530863 IC50 = 830 nM T99089 CC0WN1 155531780 IC50 = 342 nM T99089 CTMD13 155531884 IC50 = 30 nM T99089 CVQ24P 155532080 IC50 = 3210 nM T99089 CS69CA 155532132 IC50 = 1.9 nM T99089 CAB6E5 155532196 IC50 = 160 nM T99089 C6GT5Q 155533377 IC50 = 475 nM T99089 CI6B1M 155534397 IC50 = 2115 nM T99089 CKN58D 155534426 IC50 = 157 nM T99089 CH41LY 155534535 IC50 = 29 nM T99089 C0W8FZ 155534624 IC50 = 3690 nM T99089 CB9MT3 155535246 IC50 = 12.3 nM T99089 CF37GO 155535511 IC50 = 354 nM T99089 CC3ZU4 155536475 IC50 = 34.5 nM T99089 C8CK3X 155536944 IC50 = 38 nM T99089 CJ6SF9 155538658 IC50 = 303 nM T99089 C7PGF1 155539109 IC50 > 300 nM T99089 C5J8CV 155540640 IC50 = 26 nM T99089 C4R3QZ 155541552 IC50 = 2.3 nM T99089 CEJO32 155541565 IC50 = 43.7 nM T99089 C2AV3O 155541683 IC50 = 92 nM T99089 CX0J3Y 155543780 IC50 = 11.4 nM T99089 C8ZF4H 155544511 IC50 = 15700 nM T99089 C8T0MQ 155544690 IC50 = 3250 nM T99089 CY3H1I 155545239 IC50 = 348 nM T99089 C9L2CV 155546337 IC50 > 300 nM T99089 CQXE36 155547334 IC50 = 51.6 nM T99089 CB45ZE 155548916 IC50 = 34.1 nM T99089 CQF73Y 155549371 IC50 = 440 nM T99089 CHM75U 155549823 IC50 = 140 nM T99089 CG0IV2 155550125 IC50 > 300 nM T99089 C0IK8P 155550720 IC50 = 410 nM T99089 C0W7YS 155551457 IC50 > 300 nM T99089 CAH09B 155552200 IC50 = 300 nM T99089 CHE5F1 155553390 IC50 = 26800 nM T99089 C2T4PR 155553405 IC50 = 1.2 nM T99089 C30HXP 155554372 IC50 = 47 nM T99089 CD5V3C 155556809 IC50 = 13.4 nM T99089 C59PVM 155557441 IC50 > 1000 nM T99089 CP60UD 155557689 IC50 = 1700 nM T99089 CC7ES5 155557982 IC50 = 2.1 nM T99089 CBYQ06 155559698 IC50 = 237 nM T99089 CYC23K 155560669 IC50 = 700 nM T99089 C3ISX8 155560929 IC50 = 370 nM T99089 C8SP4L 155562403 IC50 > 300 nM T99089 CLU0T2 155562940 IC50 = 540 nM T99089 C81JZW 155563388 IC50 = 150 nM T99089 CQ1Y5C 155564359 IC50 = 251 nM T99089 CFOH01 155564397 IC50 = 488 nM T99089 CM47DW 155565162 IC50 > 300 nM T99089 C62CIM 155565320 IC50 = 9420 nM T99089 CSA97I 155565690 IC50 = 470.3 nM T99089 C9QAE3 155566144 IC50 = 436 nM T99089 CH3NO1 155566774 IC50 = 15.8 nM T99089 C69ICK 155567369 IC50 = 17 nM T99089 CC0DK2 155567575 IC50 = 41 nM T99089 C0E8CV 155568098 IC50 = 1050 nM T99089 C0V2MU 135398506 IC50 = 0.16 nM T99089 CR6MZ8 136030631 IC50 < 2 nM T99089 CQ5P6E 49837197 IC50 = 2.3 nM T99089 D00NWF 5730 IC50 = 230 nM T99089 D01DDB 11515006 IC50 = 7900 nM T99089 D02BXJ 46864270 IC50 = 26 nM T99089 D06QWO 14824655 IC50 > 10 ug.mL-1 T99089 D06WJA 9950176 IC50 = 10 nM T99089 D09ADW 53484100 IC50 = 0.7 nM T99089 D0A1CM 5281855 IC50 = 1760 nM T99089 D0C0ZC 11676786 IC50 < 1 nM T99089 D0D6MH 11617559 IC50 > 4800 nM T99089 D0G3SZ 6918469 IC50 = 3.3 ug.mL-1 T99089 D0GD8Y 3006531 IC50 = 250 nM T99089 D0OR5S 11631107 IC50 = 18000 nM T99089 D0OZ2S 11785878 IC50 = 540 nM T99089 D0T3PW 5281672 IC50 = 1562 nM T99089 D0Z5TQ 5924208 IC50 = 10.71 nM T23276 D0W5HK 216239 IC50 = 18.1 nM T23276 D02UFQ 11620908 IC50 > 10000 nM T23276 D05ADP 160355 IC50 = 34000 nM T23276 D0E3TC 44259 IC50 = 1310 nM T23276 D0L1GD 58282870 IC50 = 20 nM T23276 D0LF1U 5287969 IC50 = 16000 nM T23276 D0O6ZO 9952773 IC50 > 10000 nM T23276 D0Q4IX 71727581 IC50 = 1.2 nM T23276 D0X4MN 11597537 IC50 = 480 nM T23276 D0WS1V 448991 IC50 = 3300 nM T23276 D00PWQ 3820 IC50 = 20000 nM T23276 D00BPA 4592 IC50 = 25000 nM T23276 D04FHB 6918852 Ki > 50000 nM T23276 D0T3ME 156422 IC50 > 20000 nM T23276 C4MNG8 445840 IC50 > 10000 nM T23276 CVN83J 656950 IC50 > 10000 nM T23276 CDK3J0 5703619 IC50 = 1146 nM T23276 C5AL8S 6445230 EC50 = 0.55 nM T23276 CPQ13K 9933545 IC50 > 100000000 nM T23276 C0V7UW 9958506 IC50 > 11000 nM T23276 C2W3AV 9995236 IC50 > 100000 nM T23276 CV8TY1 9996476 IC50 > 10000 nM T23276 CUY0F8 10005715 IC50 > 10000 nM T23276 CF1D6Y 10075240 IC50 > 10000 nM T23276 CPS9U3 10319232 IC50 > 10000 nM T23276 CLX54H 11317348 IC50 > 10000 nM T23276 C0APW4 11422034 IC50 > 10000 nM T23276 CTG83F 11539329 Ki > 9200 nM T23276 CMIL86 11590363 Ki > 9200 nM T23276 C9T6SC 11640926 Ki > 9200 nM T23276 CJ9KN7 11683817 IC50 > 10000 nM T23276 CU0E8O 11690457 Ki > 2900 nM T23276 CB0AP2 11705863 Ki > 10000 nM T23276 CVC2S4 11722798 IC50 > 10000 nM T23276 CHR92S 11858109 IC50 > 100000 nM T23276 C7LB4I 15949613 IC50 > 10000 nM T23276 CZK8V6 16043304 IC50 = 400 nM T23276 C9TU1O 16046126 IC50 > 1000 nM T23276 CGC34R 16118737 IC50 > 100000 nM T23276 C9BI2Y 23060924 IC50 > 1100 nM T23276 C2NLE3 23060985 IC50 > 1100 nM T23276 CE7K3W 23532567 IC50 > 10000 nM T23276 CQNP54 24764449 IC50 = 100000 nM T23276 C4Z9CN 24769780 IC50 > 100000 nM T23276 CS3Q8B 24995659 IC50 > 2000 nM T23276 CTV54O 25123227 IC50 > 10000 nM T23276 C6FGQ1 25206346 IC50 > 10000 nM T23276 CU9E4P 42629114 IC50 > 10000 nM T23276 CEL61X 44229839 IC50 > 10000 nM T23276 CYE36B 44241613 IC50 > 40000 nM T23276 C6LG5T 44241614 IC50 > 40000 nM T23276 C7PRE3 44315929 IC50 = 90000 nM T23276 CUY8A3 44401410 IC50 = 300 nM T23276 C8L5ZH 44401437 IC50 > 1000 nM T23276 CIB5V1 44401506 IC50 = 750 nM T23276 C5C3BG 44401556 IC50 > 1000 nM T23276 CH0CT1 44451687 IC50 > 1100 nM T23276 C5MQX7 44451688 IC50 > 1100 nM T23276 C8K5LD 44451690 IC50 > 1100 nM T23276 C0HY3S 44451713 IC50 > 1100 nM T23276 C3VRO9 44557921 IC50 > 10000 nM T23276 C87FEM 45270051 IC50 > 40000 nM T23276 CU53FK 45273505 IC50 > 40000 nM T23276 CMB32E 46203864 IC50 = 980 nM T23276 CUA97D 46209401 IC50 > 10000 nM T23276 C60GAV 46929544 IC50 > 8000 nM T23276 CP34VL 46929748 IC50 > 1000 nM T23276 CJ2E9Q 46929857 IC50 > 25000 nM T23276 CB0S2P 49842666 IC50 > 100000 nM T23276 CAI20B 49842778 IC50 > 100000 nM T23276 CD2K4R 50908681 Ki > 1000000 nM T23276 COVJ29 50994971 IC50 = 4800 nM T23276 CEQN27 52936621 Ki > 2000 nM T23276 CD4H3S 53354074 Ki > 1000 nM T23276 C8NA4L 53384644 IC50 > 30000 nM T23276 CM8JX1 56604907 IC50 = 25000 nM T23276 CN96GA 57685722 IC50 = 207 nM T23276 CRZY38 57686268 IC50 = 25 nM T23276 CPVO76 57686351 IC50 = 43 nM T23276 CP2B1Q 57686448 IC50 = 41 nM T23276 CI19SK 57686585 IC50 = 135 nM T23276 C2ZUY5 58282827 IC50 = 7.9 nM T23276 C8MBE7 58282833 IC50 = 74 nM T23276 C1MR8Q 60097495 IC50 > 10000 nM T23276 CV63UL 67240318 IC50 > 10000 nM T23276 C1IEJ2 70789254 IC50 = 60000 nM T23276 C8T7ZP 70789255 IC50 = 37000 nM T23276 CEBO91 71452977 IC50 > 10000 nM T23276 CHQZ25 71459584 IC50 > 10000 nM T23276 CZ31PU 71583657 IC50 > 10000 nM T23276 CV4HO3 71726759 IC50 = 1070 nM T23276 C35NLY 71726760 IC50 = 150 nM T23276 C6NVW2 71726764 IC50 = 510 nM T23276 CIN10C 71727133 IC50 = 2.7 nM T23276 COI5S0 71727368 IC50 = 3.9 nM T23276 CV2CR0 71727369 IC50 = 13 nM T23276 C2XZW3 72708899 IC50 > 40000 nM T23276 CKN46T 72708901 IC50 > 40000 nM T23276 CJ2T9E 76332983 IC50 > 10000 nM T23276 C6ZSG5 84973107 IC50 = 20 nM T23276 C5VA2J 84973109 IC50 = 18 nM T23276 CP0WM3 86696674 IC50 = 7.9 nM T23276 C1O0BS 89794860 IC50 = 85 nM T23276 C54NBM 89795059 IC50 = 27 nM T23276 CYLX17 89795073 IC50 = 62 nM T23276 CO1UM8 89795095 IC50 = 9610 nM T23276 CPHT17 89795256 IC50 = 19 nM T23276 C6KBW4 89795275 IC50 = 26 nM T23276 CW5O1N 89795280 IC50 = 550 nM T23276 C15FCX 89795282 IC50 = 74 nM T23276 CN4VB6 89795308 IC50 = 3.8 nM T23276 CSK8C3 89807688 IC50 = 5 nM T23276 C6GME9 89807821 IC50 = 43 nM T23276 C0Y8ZK 91933875 IC50 > 1000 nM T23276 C2TSV7 122177851 IC50 = 65 nM T23276 CEK9S7 122177852 IC50 = 43 nM T23276 C40APN 122177853 IC50 = 20 nM T23276 CCN6F5 122177854 IC50 = 25 nM T23276 CE68SL 122177855 IC50 = 46 nM T23276 CSFJ19 122177913 IC50 = 57 nM T23276 C53NSH 122177914 IC50 = 76 nM T23276 CJD03F 122177915 IC50 = 87 nM T23276 CX8JI0 122177916 IC50 = 89 nM T23276 CJI3N8 122177917 IC50 = 95 nM T23276 CJHF98 122177918 IC50 = 23 nM T23276 CU15EY 122177919 IC50 = 32 nM T23276 CGDL13 122177920 IC50 = 89 nM T23276 CVE19K 122177921 IC50 = 23 nM T23276 CB1HF0 122177922 IC50 = 43 nM T23276 CER2Y0 122177923 IC50 = 21 nM T23276 COQ7U6 122177924 IC50 = 23 nM T23276 CV1A2F 122177925 IC50 = 24 nM T23276 CJ6RM1 122177926 IC50 = 35 nM T23276 CC13JY 122177927 IC50 = 47 nM T23276 CWM37L 123897305 IC50 = 3100 nM T23276 CQ1V6G 127045826 IC50 = 16.7 nM T23276 C6KL7C 127045928 IC50 = 74.2 nM T23276 CHK16Q 127045929 IC50 = 154 nM T23276 CF4XM2 127045932 IC50 = 78.7 nM T23276 CC9FG2 127045933 IC50 = 26.3 nM T23276 CBQ2N5 127046246 IC50 = 833 nM T23276 CLM41O 127046585 IC50 = 19.4 nM T23276 CO6Q4N 127047015 IC50 = 35.9 nM T23276 CTCR73 127047016 IC50 = 46.3 nM T23276 C6AVN3 127047018 IC50 = 29.2 nM T23276 CLG53I 127047019 IC50 = 72.4 nM T23276 CK49NV 127047027 IC50 = 53.4 nM T23276 C3WGY8 127047160 IC50 = 38.7 nM T23276 CZ3NX1 127047176 IC50 = 66.9 nM T23276 CG89KZ 127047589 IC50 = 55.5 nM T23276 CLO6T3 127047590 IC50 = 26.4 nM T23276 CY3J0C 127047591 IC50 = 29.3 nM T23276 CKQ9P4 127047724 IC50 = 22.2 nM T23276 CO6DK5 127047745 IC50 = 106 nM T23276 C0FM1R 130196825 IC50 = 13545 nM T23276 C7PS8C 135271570 IC50 = 6900 nM T23276 CG67XB 137210065 IC50 = 111 nM T23276 C0CV4B 137210066 IC50 = 32.3 nM T23276 C3FC1W 137631894 IC50 > 10000 nM T23276 C10BTW 137632556 IC50 > 10000 nM T23276 C2J9GO 137633617 IC50 > 10000 nM T23276 C7MD0H 137635615 IC50 = 790 nM T23276 CML76T 137635976 IC50 > 10000 nM T23276 CS9AW4 137636754 IC50 = 7600 nM T23276 C7R0MS 137638615 IC50 > 10000 nM T23276 CGR5B1 137642299 IC50 = 8700 nM T23276 C26HIT 137643417 IC50 > 10000 nM T23276 CDA2N6 137644922 IC50 = 278 nM T23276 CAT49C 137645403 IC50 > 10000 nM T23276 CUES49 137646218 IC50 > 10000 nM T23276 CS6J8X 137646633 IC50 > 10000 nM T23276 C9Z6NB 137646838 IC50 = 5200 nM T23276 C2HFR6 137648529 IC50 > 10000 nM T23276 CYR2I7 137649411 IC50 > 10000 nM T23276 C17GBS 137649678 IC50 > 10000 nM T23276 CEO70C 137650358 IC50 > 10000 nM T23276 C4NM0R 137650776 IC50 > 10000 nM T23276 CL3P8Q 137653011 IC50 = 7300 nM T23276 C5B9AM 137653362 IC50 = 8300 nM T23276 C8K0OY 137655533 IC50 > 10000 nM T23276 C83XOY 137657177 IC50 = 1620 nM T23276 CF7U5Y 137657487 IC50 > 10000 nM T23276 C3SD7B 137658277 IC50 > 10000 nM T23276 CVY3F0 137658568 IC50 > 10000 nM T23276 CJK81S 137659431 IC50 = 4700 nM T23276 CUS48N 137659983 IC50 > 10000 nM T23276 C6VB3O 145925651 IC50 >= 5000 nM T23276 C5TS1A 145964021 IC50 = 93 nM T23276 C8QAU0 145965069 IC50 = 952 nM T23276 CQJP12 145968722 IC50 = 45 nM T23276 CD7X3A 145969845 IC50 = 228 nM T23276 CG01BZ 145973754 IC50 = 34 nM T23276 C6X8PU 145975686 IC50 = 19 nM T23276 C28XFL 145977776 IC50 = 663 nM T23276 C2FA4R 145978301 IC50 = 17 nM T23276 CHIB04 146634736 IC50 = 21 nM T23276 C3MR9I 146634737 IC50 = 3.6 nM T23276 C6Q3UP 146634739 IC50 = 1.5 nM T23276 CX76AZ 146634741 IC50 = 4.1 nM T23276 C10WET 148308905 IC50 = 3.3 nM T23276 C86HPW 155518524 IC50 = 65000 nM T23276 D00HVA 11624601 Ki > 9200 nM T23276 D01MNK 25125014 IC50 = 3730 nM T23276 D02XHC 448912 IC50 = 18000 nM T23276 D04PEI 11467730 IC50 > 50000 nM T23276 D07OAT 456214 IC50 = 9000 nM T23276 D07OXC 11650194 IC50 > 100000 nM T23276 D08XVZ 24866313 IC50 = 4 nM T23276 D09RYV 9911652 IC50 > 100000000 nM T23276 D0OZ2S 11785878 IC50 > 100000 nM T23276 D0Q3NG 11715520 Ki > 9200 nM T23276 D0S7IE 11658882 Ki > 9200 nM T23276 D0UN9O 3385203 IC50 >= 10000 nM T23276 D0V0QJ 389898 IC50 = 82900 nM T23276 D0ZG4G 11493598 Ki = 310 nM T85616 D04JTD 219104 IC50 = 2110 nM T85616 CI7MW0 9852185 Ki = 3110 nM T85616 C5DL2O 15335087 IC50 = 510 nM T85616 C6W2MC 71487261 IC50 = 340 nM T85616 CB52OT 71487263 IC50 = 7310 nM T85616 CJC7Y6 71562811 IC50 = 170 nM T85616 CM1VW2 71562812 IC50 = 90 nM T85616 CG3U8R 71562814 IC50 = 240 nM T85616 C6VPK1 71562930 IC50 = 450 nM T85616 CU35ZW 71562931 IC50 = 540 nM T85616 CBM95V 136240922 IC50 = 290 nM T81503 D0Q0PR 54675769 IC50 = 154 nM T81503 CLQ19N 54695811 IC50 = 43 nM T81503 CJ4Q5C 54695812 IC50 = 137 nM T81503 CN2LR7 54695813 IC50 = 276 nM T81503 CWGP52 54697399 IC50 = 75 nM T81503 CWL92P 54708659 IC50 = 22 nM T81503 C0QL6P 54713406 IC50 = 891 nM T81503 C50NPL 54721832 IC50 = 131 nM T81503 C94HJN 54729434 IC50 > 10000 nM T81503 CNQI70 54729435 IC50 = 17 nM T81503 CK9Q2M 54729436 IC50 = 86 nM T81503 C6ECK7 54729437 IC50 = 219 nM T81503 CU04CO 54729438 IC50 = 140 nM T81503 C0T2FR 54729439 IC50 = 190 nM T81503 C9F2HC 54729448 IC50 > 10000 nM T81503 CG90ET 54729449 IC50 > 10000 nM T81503 CI78JU 54729450 IC50 = 20 nM T81503 C30HTF 54729451 IC50 = 116 nM T81503 CFWS93 54729452 IC50 = 110 nM T81503 CEA05G 54730369 IC50 = 34 nM T81503 CI1SU0 54730370 IC50 = 280 nM T81503 CIE25B 54730375 IC50 > 10000 nM T81503 C8ZM7I 54730379 IC50 = 41 nM T81503 C1E4WO 54730380 IC50 = 106 nM T81503 C73YWX 54730381 IC50 = 320 nM T81503 C6C1KM 54730382 IC50 = 598 nM T81503 CD2P1F 54732401 IC50 < 5 nM T81503 CMIN96 54732402 IC50 = 44 nM T81503 CR9TB4 54732403 IC50 = 460 nM T81503 CG92WX 54732408 IC50 > 10000 nM T81503 C4GHD2 54732409 IC50 = 19 nM T81503 CHGE48 54732410 IC50 = 120 nM T81503 D0C9BH 54706138 IC50 < 5 nM T33492 D04NDM 165580 IC50 = 21000000 nM T33492 D05JNI 8378 IC50 = 8000000 nM T33492 D07JZF 441306 IC50 = 8000000 nM T33492 D0GZ7B 5328779 IC50 > 333000 nM T33492 CI26AQ 1607 IC50 = 360 nM T33492 C5IF7O 2259 IC50 = 12 nM T33492 CW68ZS 61672 IC50 = 4000 nM T33492 CYTJ80 78402 IC50 > 10000 nM T33492 CH67EZ 91286 IC50 > 111000 nM T33492 C0O3TQ 126437 IC50 = 1230 nM T33492 CH6PG4 203854 IC50 > 10000 nM T33492 CZTD26 220436 IC50 > 111000 nM T33492 C80UDV 334474 IC50 > 111000 nM T33492 CS2B8E 397888 IC50 = 12000 nM T33492 CESM72 439530 IC50 = 18000000 nM T33492 C0KE3R 442614 IC50 > 100000 nM T33492 CX9UA1 443385 IC50 = 9100000 nM T33492 CX8VI4 561354 IC50 = 9170 nM T33492 C34CEH 676561 IC50 = 710 nM T33492 C2Z0SV 685482 IC50 > 333000 nM T33492 CAPG06 726820 IC50 > 333000 nM T33492 C9NYF1 728520 IC50 = 5280 nM T33492 CF32MI 766914 IC50 > 333000 nM T33492 CE10WO 776842 IC50 = 110 nM T33492 C18SJQ 885337 IC50 > 10000 nM T33492 C2P9DB 1005270 IC50 > 15000 nM T33492 C47QWD 1025279 IC50 = 1000 nM T33492 C13SDI 1115047 IC50 = 500 nM T33492 CSO84U 1188215 IC50 > 10000 nM T33492 CBG3X5 1236521 IC50 = 40000 nM T33492 C2REL7 1239884 IC50 > 333000 nM T33492 C0SKV6 1325590 IC50 > 10000 nM T33492 CIZ70U 1325673 IC50 > 10000 nM T33492 CLA9J7 1540149 IC50 = 34000 nM T33492 CU5PF6 1652110 IC50 > 333000 nM T33492 CRL05A 1771058 IC50 = 7700 nM T33492 CP31XF 2030903 IC50 = 4930 nM T33492 C8WS4M 2040507 IC50 > 10000 nM T33492 CQI6S5 2243892 IC50 = 111000 nM T33492 C80CJH 2441756 IC50 = 14130 nM T33492 CAT8Q3 3000500 IC50 = 8000000 nM T33492 CI34YK 3121217 IC50 = 5620 nM T33492 C4N0CE 5328793 IC50 > 333000 nM T33492 C48BJI 5336179 IC50 = 1080 nM T33492 C3YD4V 5351985 IC50 = 14000 nM T33492 CX30RB 5411062 IC50 > 333000 nM T33492 CO01XP 5478021 IC50 > 111000 nM T33492 C26DVM 6211778 IC50 > 333000 nM T33492 C5PT6B 6245483 IC50 > 111000 nM T33492 CO6J1X 6304702 IC50 = 12000 nM T33492 C2MZ9A 7083198 IC50 = 950 nM T33492 CL6Z8O 7454864 IC50 = 19000 nM T33492 C6XP2L 9139208 IC50 = 35480 nM T33492 CO5Q7F 10338255 IC50 = 22300 nM T33492 CRBZ37 10494779 IC50 > 111000 nM T33492 C0YD4S 10640393 IC50 > 111000 nM T33492 CG07YZ 10663416 IC50 > 111000 nM T33492 CIO2Y3 11220435 Ki = 3190 nM T33492 C5F6NY 11370831 IC50 = 55300 nM T33492 CBU10H 11520588 IC50 = 1000 nM T33492 CRS8D5 12525013 IC50 = 30000 nM T33492 CT91GZ 16098813 IC50 = 5800 nM T33492 CKZ5B8 16098830 IC50 = 1000 nM T33492 CV8TP1 16221202 IC50 = 17500 nM T33492 CJ32LD 16221204 IC50 = 31000 nM T33492 CFD49E 16221206 IC50 = 47000 nM T33492 C17EIS 16221208 IC50 = 14100 nM T33492 C1MRB8 16221210 IC50 = 33000 nM T33492 CT32AS 16221263 IC50 = 25000 nM T33492 C67THG 16221322 IC50 = 48000 nM T33492 CIW39K 16221324 IC50 = 14100 nM T33492 CO42ZD 16434867 IC50 = 50120 nM T33492 CE0Q5Z 17390511 IC50 = 44000 nM T33492 CX30ZC 17756086 IC50 = 37000 nM T33492 C4KUW5 18230892 IC50 = 79430 nM T33492 C2RSJ0 41587290 IC50 = 11220 nM T33492 C7UM4C 42630956 IC50 = 27000 nM T33492 CD97JI 42915055 IC50 = 44670 nM T33492 CZQN61 44574209 IC50 = 1800000 nM T33492 CF48PX 45353287 IC50 = 44670 nM T33492 C9VHP4 46229345 IC50 = 35000 nM T33492 C92NHR 46229346 IC50 = 5000 nM T33492 CCM26J 56837840 IC50 > 111000 nM T33492 CPA1M7 57521375 IC50 > 111000 nM T33492 C98GSX 57521376 IC50 > 111000 nM T33492 C6UIY2 57521377 IC50 > 111000 nM T33492 C3V0GK 57521378 IC50 > 111000 nM T33492 CX82UH 57521379 IC50 > 111000 nM T33492 C13AUV 57521485 IC50 > 111000 nM T33492 CRZ52K 57521486 IC50 > 111000 nM T33492 C0UT7F 57521488 IC50 > 111000 nM T33492 C7ID1U 57521489 IC50 > 111000 nM T33492 CQK0F8 57521585 IC50 > 111000 nM T33492 CM8VZ1 57521586 IC50 > 111000 nM T33492 C13XAL 57521587 IC50 > 111000 nM T33492 C9HV4M 57521588 IC50 > 111000 nM T33492 C3U9EO 57521589 IC50 > 111000 nM T33492 CN72YQ 57521691 IC50 > 111000 nM T33492 C3AXR7 57521692 IC50 > 111000 nM T33492 C4FIE9 57521693 IC50 > 111000 nM T33492 CR38GS 57521694 IC50 > 111000 nM T33492 C6CUL8 57521695 IC50 > 111000 nM T33492 CJ6Z3M 57521803 IC50 > 111000 nM T33492 CG5YJ9 57521804 IC50 > 111000 nM T33492 C5E6VB 57521805 IC50 > 111000 nM T33492 CB1E5V 57521806 IC50 > 111000 nM T33492 C1L0TI 57521807 IC50 > 111000 nM T33492 CP36UT 57521909 IC50 > 111000 nM T33492 C4HP8U 57521910 IC50 > 111000 nM T33492 CQV97O 57521911 IC50 > 111000 nM T33492 CYO01C 57521912 IC50 > 111000 nM T33492 C7VBQ4 57522032 IC50 > 111000 nM T33492 C8J3FI 57522033 IC50 > 111000 nM T33492 CB3L2W 57522034 IC50 > 111000 nM T33492 CTO5S8 57522035 IC50 > 111000 nM T33492 CTRX83 57522599 IC50 > 111000 nM T33492 CRP57E 57522600 IC50 > 111000 nM T33492 CQUG46 57522601 IC50 > 111000 nM T33492 CIJ19L 57522602 IC50 > 111000 nM T33492 C6DC1K 57522711 IC50 > 111000 nM T33492 CB9OC3 57522712 IC50 > 111000 nM T33492 CN7Q3O 57522716 IC50 > 111000 nM T33492 CP2LO3 57522717 IC50 > 111000 nM T33492 CUA7L4 57522821 IC50 > 111000 nM T33492 CW31RU 57522822 IC50 > 111000 nM T33492 CPOR59 57522823 IC50 > 111000 nM T33492 CJA90N 57522824 IC50 > 111000 nM T33492 CBSY92 57522825 IC50 > 111000 nM T33492 C0QLK6 57522826 IC50 > 111000 nM T33492 C3BI1S 57522959 IC50 > 111000 nM T33492 CNF76K 57522960 IC50 > 111000 nM T33492 CWL8R4 57522961 IC50 > 111000 nM T33492 CIL52C 57522962 IC50 > 111000 nM T33492 C09IFB 57522963 IC50 > 111000 nM T33492 CTP92I 57522964 IC50 > 111000 nM T33492 CQ97US 57523098 IC50 > 111000 nM T33492 CQ82LU 57523099 IC50 > 111000 nM T33492 C08FVX 57523100 IC50 > 111000 nM T33492 C5CQT0 57523101 IC50 > 111000 nM T33492 CAF3X4 57523102 IC50 > 111000 nM T33492 C6AZ0X 60148508 IC50 = 12000 nM T33492 CO4P2S 60148514 IC50 = 37000 nM T33492 CH95XR 60165808 IC50 = 18000 nM T33492 C1Q7GJ 60165957 IC50 > 111000 nM T33492 CQZ2N7 60165960 IC50 > 111000 nM T33492 CMW7P2 60165963 IC50 > 111000 nM T33492 CHW9Y7 60166112 IC50 > 111000 nM T33492 CNF46Y 66489030 IC50 = 26000 nM T33492 CB6A5C 70674149 IC50 > 10000 nM T33492 CXAT75 70690590 IC50 > 111000 nM T33492 CWU83Q 70696734 IC50 > 111000 nM T33492 C9M8FA 71449815 IC50 > 333000 nM T33492 CA71WP 71450009 IC50 = 37000 nM T33492 C5VT8U 71451618 IC50 = 11000 nM T33492 CHW4O9 71451620 IC50 = 15000 nM T33492 CX6JV8 71451621 IC50 = 46000 nM T33492 CYI5H3 71451622 IC50 = 20000 nM T33492 CJ68NX 71451623 IC50 = 69000 nM T33492 CP3FA6 71451624 IC50 = 74000 nM T33492 C9CUO8 71452527 IC50 = 1620 nM T33492 CAJ47F 71452528 IC50 = 260 nM T33492 CHD2O4 71453458 IC50 = 8500 nM T33492 CJ83PN 71453459 IC50 = 138000 nM T33492 C69BNH 71453460 IC50 = 13000 nM T33492 CXM5V1 71453461 IC50 > 333000 nM T33492 CI6O5J 71453649 IC50 > 111000 nM T33492 C51XKH 71454291 IC50 = 1540 nM T33492 C4TWY0 71455170 IC50 = 75000 nM T33492 C34SCA 71456960 IC50 = 6900 nM T33492 C7FPV4 71456961 IC50 = 34000 nM T33492 C4VO0K 71456962 IC50 > 333000 nM T33492 CZ3K8E 71457146 IC50 > 111000 nM T33492 CN4CR6 71458831 IC50 = 51000 nM T33492 CCLK82 71458832 IC50 = 111000 nM T33492 CX9SE4 71460811 IC50 > 111000 nM T33492 CRT0H9 71461477 IC50 = 940 nM T33492 C1H3AJ 71461478 IC50 = 1810 nM T33492 CHCX75 71461479 IC50 = 570 nM T33492 CIM47J 71462348 IC50 = 38000 nM T33492 C9D6YL 71462349 IC50 = 28000 nM T33492 CBHZ04 71462352 IC50 = 29000 nM T33492 C04MQY 71544698 IC50 > 111000 nM T33492 CXY45D 71544701 IC50 > 111000 nM T33492 C6SZ7F 71544702 IC50 > 111000 nM T33492 C3ARJ0 71544866 IC50 = 12000 nM T33492 CBOR04 71544868 IC50 > 111000 nM T33492 CG3VH5 71545025 IC50 = 5200 nM T33492 C7KLX0 71545027 IC50 = 6700 nM T33492 CZ7NG2 71546175 IC50 > 111000 nM T33492 CEM9V0 71546176 IC50 > 111000 nM T33492 CS7ZY0 71546177 IC50 > 111000 nM T33492 CKJ42V 71546178 IC50 > 111000 nM T33492 C9JI8X 71546179 IC50 > 111000 nM T33492 CA49VP 71546347 IC50 = 61000 nM T33492 C7R0VX 71546348 IC50 > 111000 nM T33492 C7NIU6 71546350 IC50 > 111000 nM T33492 CTA72F 71546351 IC50 > 111000 nM T33492 C3B2LW 71546514 IC50 > 111000 nM T33492 C4WZ3O 71546516 IC50 = 45000 nM T33492 CYL3F6 71546517 IC50 = 18000 nM T33492 CTI3N1 71546518 IC50 = 37000 nM T33492 CK0C3J 71546671 IC50 = 37000 nM T33492 CZ49YE 71546672 IC50 = 37000 nM T33492 CH46SD 71546675 IC50 = 37000 nM T33492 C1Z0GN 71546826 IC50 > 111000 nM T33492 CDA9V1 71546829 IC50 > 111000 nM T33492 C1VIY2 71546831 IC50 > 111000 nM T33492 C9Q4YR 71546833 IC50 > 111000 nM T33492 C3Y9MP 71546979 IC50 > 111000 nM T33492 C41YVT 71546981 IC50 > 111000 nM T33492 C28KSH 71546982 IC50 > 111000 nM T33492 C4MSG0 71546985 IC50 = 11000 nM T33492 C7U1WD 71546986 IC50 > 111000 nM T33492 C1O5HY 71547124 IC50 > 111000 nM T33492 C7VJN5 71547126 IC50 = 5000 nM T33492 C3GPU9 71547128 IC50 > 111000 nM T33492 CO38NF 71547129 IC50 > 111000 nM T33492 C9Q4DA 71547131 IC50 = 15000 nM T33492 CVS84W 71582100 IC50 = 3800 nM T33492 C94DIL 73334714 IC50 > 111000 nM T33492 CRZ62F 73355036 IC50 = 5000 nM T33492 CMU46W 76029213 IC50 > 111000 nM T33492 CA4F7D 76311078 IC50 > 111000 nM T33492 C40TDU 76311079 IC50 > 111000 nM T33492 CF08AN 76311080 IC50 > 111000 nM T33492 CT05OM 76311081 IC50 = 37000 nM T33492 C24IZB 76311082 IC50 = 12000 nM T33492 CC84YZ 76314698 IC50 = 37000 nM T33492 CTQW89 76314699 IC50 > 111000 nM T33492 CVN17S 76318268 IC50 > 111000 nM T33492 C32WVQ 76318269 IC50 > 111000 nM T33492 C9KN5G 76318270 IC50 = 37000 nM T33492 C9Y0MW 76321973 IC50 > 111000 nM T33492 CF24IO 76321974 IC50 > 111000 nM T33492 C8NP5E 76329155 IC50 > 111000 nM T33492 CE8A1M 76329156 IC50 = 37000 nM T33492 C8WB7V 76332814 IC50 > 111000 nM T33492 CL3QN6 76332815 IC50 = 37000 nM T33492 CJSL58 76332816 IC50 = 12000 nM T33492 C3D6MK 76336438 IC50 = 37000 nM T33492 CB6YU7 86291808 IC50 = 5500 nM T33492 C6JV2S 86765191 IC50 = 12000 nM T33492 CQU1J7 86765192 IC50 = 12000 nM T33492 C30VXB 86765193 IC50 > 111000 nM T33492 CK1Y4C 86765194 IC50 = 12000 nM T33492 CN64AH 86765195 IC50 = 1000 nM T33492 C9NV1H 86765208 IC50 > 111000 nM T33492 CT6YB9 90643550 IC50 > 111000 nM T33492 C3LS5W 90643551 IC50 > 111000 nM T33492 CDQG63 90643552 IC50 > 111000 nM T33492 CH25QC 90643553 IC50 = 37000 nM T33492 C8QC2J 110206286 IC50 = 790 nM T33492 C4WE5F 110207923 IC50 = 1530 nM T33492 CUVY69 118070452 IC50 = 37000 nM T33492 CG94AY 118070454 IC50 = 12000 nM T33492 CFQ3A4 118721722 IC50 = 390 nM T33492 C5M8NJ 118721723 IC50 = 150 nM T33492 CFP6G9 118721724 IC50 = 810 nM T33492 C3ZOW1 118721725 IC50 = 450 nM T33492 C9JEB8 118727325 IC50 > 10000 nM T33492 CVL96K 118728738 IC50 = 3700 nM T33492 CVWY39 118728739 IC50 = 1280 nM T33492 CC42ZN 118728740 IC50 = 1620 nM T33492 C8N0QE 118728741 IC50 = 220 nM T33492 CNH9E7 118728742 IC50 = 6030 nM T33492 C65CJL 118728743 IC50 = 3660 nM T33492 CK2C9Z 118728744 IC50 = 1300 nM T33492 CJ3C4L 118735563 IC50 > 111000 nM T33492 CBZF47 118735565 IC50 > 111000 nM T33492 CUN56B 118735568 IC50 > 111000 nM T33492 CQC6B9 118735570 IC50 = 12000 nM T33492 CYIM15 118735572 IC50 = 12000 nM T33492 C6GZL3 118735573 IC50 > 111000 nM T33492 CCA73K 118735574 IC50 > 111000 nM T33492 CTN0Y6 118735576 IC50 = 12000 nM T33492 CDC9A2 118735578 IC50 > 111000 nM T33492 CXB0R3 118735580 IC50 > 111000 nM T33492 CP1W7A 118735582 IC50 = 1000 nM T33492 C46INW 118735583 IC50 > 111000 nM T33492 CXJG20 118735584 IC50 > 111000 nM T33492 CGN27Z 118735585 IC50 = 37000 nM T33492 CFKO57 118735587 IC50 > 111000 nM T33492 CR7UK8 118735588 IC50 > 111000 nM T33492 CU0KP6 118735590 IC50 = 12000 nM T33492 CH30JX 121478365 IC50 = 38000 nM T33492 CT1RL3 122179149 IC50 > 111000 nM T33492 CM9AU7 122179162 IC50 > 111000 nM T33492 C98KOJ 122179163 IC50 = 63000 nM T33492 C7Q9FC 122179164 IC50 > 111000 nM T33492 CY2Q4V 122181724 IC50 = 1000 nM T33492 CK91CX 122181725 IC50 = 1000 nM T33492 CG3O5N 122483604 IC50 > 111000 nM T33492 C7BL9T 122484905 IC50 = 6200 nM T33492 C3FS6Y 122484906 IC50 = 6300 nM T33492 CS1DF2 127025946 IC50 = 1700 nM T33492 CG8BR2 127028127 IC50 = 2200 nM T33492 CLT35C 127043728 IC50 > 111000 nM T33492 CJA2I1 127044083 IC50 = 63000 nM T33492 CBFS34 127044239 IC50 > 111000 nM T33492 CE15TB 127044402 IC50 > 111000 nM T33492 CF64IU 127044403 IC50 > 111000 nM T33492 C12IUQ 127044404 IC50 = 90000 nM T33492 CBE49O 127044405 IC50 > 111000 nM T33492 CM19WU 127044406 IC50 = 19000 nM T33492 CU15SD 127044408 IC50 > 111000 nM T33492 C0X5YU 127044409 IC50 = 30000 nM T33492 C3XO0J 127044411 IC50 > 111000 nM T33492 COX07F 127044412 IC50 = 111000 nM T33492 C5OQ3T 127044413 IC50 > 111000 nM T33492 C38YZG 127044414 IC50 > 60000 nM T33492 C0SP4E 127044557 IC50 = 43000 nM T33492 CPEU65 127044559 IC50 > 111000 nM T33492 C1W8YR 127044560 IC50 > 111000 nM T33492 C4ZI7L 129751977 IC50 = 1010 nM T33492 C8TM2K 129881957 IC50 = 190 nM T33492 CP7E6T 129881996 IC50 = 160 nM T33492 C72SJL 129883811 IC50 = 4100 nM T33492 C0C7LT 129883861 IC50 = 1250 nM T33492 CYI8M7 129883900 IC50 = 1210 nM T33492 C6X7VK 129883904 IC50 = 610 nM T33492 CRK13E 129883976 IC50 = 1120 nM T33492 CVE65K 129884019 IC50 = 5900 nM T33492 C9L1GO 129896914 IC50 = 1000 nM T33492 C2BV6U 132577626 IC50 = 1390 nM T33492 C6JL5C 132577627 IC50 = 1920 nM T33492 C6DQL0 132577629 IC50 = 750 nM T33492 C94PEK 134132337 IC50 = 675 nM T33492 C1BN0D 134135136 IC50 = 4310 nM T33492 CU50NE 134138761 IC50 = 1230 nM T33492 C3AJ4Y 134140308 IC50 = 1200 nM T33492 C4W5YX 134140937 IC50 = 1370 nM T33492 CVH14W 134142079 IC50 = 1450 nM T33492 C9KZI1 134150902 IC50 = 1560 nM T33492 CE49RL 134156830 IC50 = 1090 nM T33492 C5DA0Z 135163962 IC50 = 12000 nM T33492 CC57MQ 135400994 IC50 = 18000 nM T33492 C7PO0L 135541470 IC50 > 111000 nM T33492 CS8HM5 135815232 IC50 = 11000 nM T33492 C1R7MT 135875770 IC50 = 111000 nM T33492 CVR0T7 136236290 IC50 = 48000 nM T33492 CTG7U8 136236291 IC50 = 39000 nM T33492 C5K9YU 136236292 IC50 = 35000 nM T33492 CLEM70 136236293 IC50 = 7100 nM T33492 C04RXQ 136236294 IC50 = 4100 nM T33492 CEBA65 136236295 IC50 = 220000 nM T33492 CN0VR1 136236296 IC50 = 12000 nM T33492 CF7M6P 136236297 IC50 = 2600 nM T33492 C8EZC7 136236298 IC50 = 111000 nM T33492 CR31TD 136236299 IC50 = 111000 nM T33492 CNIM68 136236300 IC50 = 32000 nM T33492 CQZ79S 137633472 IC50 > 111000 nM T33492 CEMW84 137634763 IC50 = 1000 nM T33492 CY83RB 137635101 IC50 > 111000 nM T33492 CY4BH7 137635982 IC50 = 12000 nM T33492 CP8I0N 137635992 IC50 > 111000 nM T33492 CC1X7N 137637372 IC50 = 33300 nM T33492 CSKE17 137638583 IC50 = 27500 nM T33492 C7K5XB 137638718 IC50 > 111000 nM T33492 CY0G2M 137639745 IC50 = 11900 nM T33492 CE93VQ 137639878 IC50 > 111000 nM T33492 C7KVT8 137640123 IC50 = 1000 nM T33492 CT5YB3 137641552 IC50 > 100000 nM T33492 C7EHL1 137643195 IC50 > 111000 nM T33492 CQ89WF 137644721 IC50 = 20200 nM T33492 C7LY3U 137645346 IC50 = 14000 nM T33492 CT8A6V 137645479 IC50 = 1000 nM T33492 CTD0Q1 137645708 IC50 = 12000 nM T33492 C83FEH 137646143 IC50 > 111000 nM T33492 CR72BP 137646560 IC50 = 12000 nM T33492 CW24CA 137650951 IC50 = 16000 nM T33492 C2MP3A 137650968 IC50 = 1000 nM T33492 C2RVW9 137651075 IC50 = 22200 nM T33492 C7SUD6 137652086 IC50 > 111000 nM T33492 C9X2IG 137652438 IC50 > 111000 nM T33492 CY25WR 137653301 IC50 > 111000 nM T33492 CDQ41E 137656446 IC50 > 111000 nM T33492 CZX8J7 137658040 IC50 > 100000 nM T33492 CZ01OK 137658578 IC50 = 1000 nM T33492 CHXA46 137659333 IC50 = 12000 nM T33492 CB9GY3 137660083 IC50 > 111000 nM T33492 C09XQR 137661166 IC50 > 111000 nM T33492 CM78PY 138454772 IC50 = 7000 nM T33492 C6KZP1 139593958 IC50 = 63 nM T33492 C81WPC 139593986 IC50 = 26 nM T33492 CDU5H3 145949386 IC50 = 13000 nM T33492 CRS2C9 145949970 IC50 = 15000 nM T33492 CDM0W7 145951675 IC50 = 48000 nM T33492 CN16JZ 145951972 IC50 = 16000 nM T33492 CO8TH1 145954631 IC50 = 20000 nM T33492 CF90QJ 145956398 IC50 = 40000 nM T33492 C8Q5BD 145960258 IC50 = 20000 nM T33492 CK83GM 145982803 IC50 = 160 nM T33492 C2WO8C 145982960 IC50 = 630 nM T33492 CS9L5D 145983163 IC50 = 64 nM T33492 CE2A0Q 145983563 IC50 = 3300 nM T33492 C61ZPL 145983762 IC50 = 980 nM T33492 CVQ4G0 145983767 IC50 = 3650 nM T33492 C5M2JX 145983887 IC50 = 230 nM T33492 C7Z4HY 145984004 IC50 = 81 nM T33492 C7SE0X 145984229 IC50 = 600 nM T33492 CT8P1S 145984246 IC50 = 340 nM T33492 CE0N3L 145984315 IC50 = 6730 nM T33492 C5IJN8 145984662 IC50 = 720 nM T33492 C0W3ZP 145985218 IC50 = 1590 nM T33492 CF8U0M 145985434 IC50 = 860 nM T33492 C95TOG 145985558 IC50 = 900 nM T33492 CZVU04 145985759 IC50 > 15000 nM T33492 CA2R9X 145985836 IC50 = 340 nM T33492 CUJ6W5 145985887 IC50 = 840 nM T33492 C7FIS3 145985899 IC50 = 1220 nM T33492 CPI14D 145985918 IC50 = 530 nM T33492 C9E1BP 145985980 IC50 = 25 nM T33492 CX4R2M 145986039 IC50 = 232 nM T33492 CSV38F 145986188 IC50 = 1020 nM T33492 C7JP2N 151276071 IC50 = 100 nM T33492 CN5B4U 155510460 IC50 = 710 nM T33492 CCP8V7 155511883 IC50 = 90 nM T33492 CV69GT 155511965 IC50 = 192 nM T33492 C3PQ4I 155514436 IC50 = 68 nM T33492 CGT9M7 155514788 IC50 = 35 nM T33492 CTFA82 155515608 IC50 = 110 nM T33492 CZ2AH9 155518351 IC50 = 158 nM T33492 CF5NE1 155519048 IC50 = 34100 nM T33492 C3BZS7 155522234 IC50 = 3500 nM T33492 C1XC9R 155525490 IC50 = 12100 nM T33492 C2C8QK 155527697 IC50 = 500 nM T33492 CK4F1S 155530696 IC50 = 5 nM T33492 C9JQ5R 155532411 IC50 = 190 nM T33492 CP7IM4 155537726 IC50 = 150 nM T33492 C0T8MV 155547340 IC50 = 457 nM T33492 CR06HT 155549764 IC50 = 3700 nM T33492 C3RC9M 155551925 IC50 = 1490 nM T33492 C0F9WC 155554203 IC50 = 2300 nM T33492 CD5NV9 155555272 IC50 = 172 nM T33492 CZU1M4 155562716 IC50 = 22 nM T33492 C4LXT8 155564630 IC50 = 570 nM T33492 C9B1AO 155566616 IC50 = 86 nM T33492 D01NTW 5328768 IC50 > 333000 nM T33492 D02BUW 2061 IC50 > 333000 nM T33492 D07SQW 72394 IC50 = 30000000 nM T33492 D09KUE 259210 IC50 = 1000 nM T33492 D0Q3GG 667601 IC50 = 12000 nM T72881 D00QET 5281040 IC50 < 5000 nM T72881 D05MCS 44473151 IC50 = 36000 nM T72881 CUF65V 2261273 IC50 = 1900 nM T72881 C79DVG 56589615 IC50 > 3000 nM T72881 CU86FL 58034959 IC50 = 35 nM T72881 CW19CN 122670086 IC50 = 7.8 nM T72881 CO81KV 122670103 IC50 = 0.66 nM T72881 C86VYP 122670110 IC50 = 0.28 nM T72881 CK2B0J 138857937 IC50 = 2.4 nM T72881 CU95NM 145983649 IC50 = 6190 nM T72881 C76ACJ 145985137 IC50 = 30 nM T72881 CM62SF 145985303 IC50 = 15860 nM T72881 CN8G1X 145993375 IC50 = 1800 nM T72881 CS27OA 150767852 IC50 = 16 nM T72881 C0O7RL 155513699 IC50 = 8.65 nM T72881 CU56QS 155514039 IC50 = 7.9 nM T72881 C03QFT 155514291 IC50 = 27.4 nM T72881 CV7H9X 155514523 IC50 = 158 nM T72881 CGE90A 155515058 IC50 = 0.758 nM T72881 CL9QK7 155515277 IC50 = 27.7 nM T72881 CVI2D6 155518247 IC50 = 11.5 nM T72881 C3LC2H 155523754 IC50 = 1.41 nM T72881 C7XH4U 155525620 IC50 = 15.5 nM T72881 CRY0J2 155530520 IC50 = 0.381 nM T72881 CYB6A8 155531199 IC50 = 24.3 nM T72881 CC62BH 155532184 IC50 = 31.8 nM T72881 C15UYV 155532743 IC50 = 3.71 nM T72881 C3IXY0 155538051 IC50 = 1.05 nM T72881 C7O4TV 155543878 IC50 = 0.36 nM T72881 C3LK0J 155544798 IC50 = 6.42 nM T72881 CI6UZ9 155546599 IC50 = 13 nM T72881 C5VU2K 155550738 IC50 = 0.28 nM T72881 C6WCU9 155552988 IC50 = 1.97 nM T72881 CHI4B5 155553658 IC50 = 14 nM T72881 CIAY61 155553929 IC50 = 5.26 nM T72881 CZH04D 155559637 IC50 = 7.09 nM T72881 CXE0N3 155560141 IC50 = 109 nM T72881 CWYM30 155560185 IC50 = 157 nM T72881 C6K3MC 155564144 IC50 = 4.74 nM T72881 CBWQ63 155564396 IC50 = 8.5 nM T72881 C5QYB7 155565891 IC50 = 0.63 nM T30081 D01XYJ 35370 Ki = 2900 nM T30081 D03TGJ 5282192 IC50 > 500000 nM T30081 D07XSN 6253 IC50 > 1000000 nM T30081 D0Z8EX 18283 Ki = 580000 nM T30081 D06CCR 50313 Ki = 140 nM T30081 D0TJ9S 445212 Ki = 16100 nM T30081 D0Z9LP 446727 Ki = 100 nM T30081 CP25DX 65049 IC50 > 1000000 nM T30081 CD85ZQ 65159 Ki = 445000 nM T30081 CO4UY8 72230 Ki = 425000 nM T30081 CO15BF 72327 Ki = 180 nM T30081 CRM8J6 162419 IC50 = 14000 nM T30081 CVZ48I 174316 Ki = 90 nM T30081 CVDG62 452392 IC50 = 44000 nM T30081 CPJ56E 452395 IC50 = 53000 nM T30081 C93KDB 459905 Ki = 210 nM T30081 C5FS1E 477012 Ki = 1040000 nM T30081 CI0S8N 477015 Ki = 970000 nM T30081 CUW3B2 491807 IC50 > 1000000 nM T30081 C8WS5I 491808 IC50 > 1000000 nM T30081 CYTV93 491811 IC50 > 1000000 nM T30081 C71RDP 497634 IC50 = 3100 nM T30081 CX2LN9 497636 IC50 = 1200 nM T30081 CLI98Q 497637 IC50 = 3300 nM T30081 CS78DH 504626 IC50 > 500000 nM T30081 CO93FT 506492 IC50 = 73000 nM T30081 CN4A5U 508215 Ki = 220000 nM T30081 CZCE20 508216 Ki = 110000 nM T30081 CO9RJ8 510135 Ki = 40000 nM T30081 CNX65O 514178 IC50 = 7800 nM T30081 C3LE1J 3000238 Ki = 1690000 nM T30081 CC8TV9 3000253 Ki = 1600000 nM T30081 CVO3D5 3000254 Ki = 54000 nM T30081 C04TFN 3000255 Ki = 1690000 nM T30081 CG1QZ5 3000256 Ki = 1275000 nM T30081 CZF20L 3006428 Ki = 32000 nM T30081 CW0B1Q 3006429 Ki = 4700 nM T30081 CB1UY3 3006430 Ki = 43500 nM T30081 CMY59Q 3006432 Ki = 280000 nM T30081 C3KGQ8 3007847 Ki = 2000 nM T30081 CETR09 3034569 Ki = 12000 nM T30081 CW15OC 6439190 Ki = 220 nM T30081 CA89BP 6476766 IC50 > 1000000 nM T30081 CJB97H 6476767 IC50 > 1000000 nM T30081 C59CWM 6477687 IC50 = 3000 nM T30081 CH7M6L 6477690 IC50 = 9800 nM T30081 C2OH8G 6477696 IC50 = 22000 nM T30081 C1BF5V 9837976 Ki = 420000 nM T30081 C5O8EM 9906078 Ki = 62900 nM T30081 CBM0K2 9971180 IC50 = 57000 nM T30081 CHNO31 10003208 IC50 = 2300 nM T30081 CQ26PR 10040442 IC50 = 30000 nM T30081 CZ1A0R 10097595 IC50 > 1000000 nM T30081 C3EF4R 10198687 Ki = 2900 nM T30081 CT9JP4 10269114 IC50 > 500000 nM T30081 CM2L4O 10406438 Ki = 85800 nM T30081 C2G4OQ 10978846 IC50 = 40000 nM T30081 C82JAI 11438492 Ki = 69800 nM T30081 C8HVL6 11825312 IC50 = 4600 nM T30081 CG5E1H 11827046 IC50 = 2 nM T30081 C2KNL5 14308783 Ki = 975000 nM T30081 C0PHT1 14606828 IC50 = 99000 nM T30081 C7W9FV 15227900 IC50 > 50000 nM T30081 C2Z9KL 15227901 IC50 = 50000 nM T30081 C6Q3KN 15227902 IC50 > 50000 nM T30081 CG1D2I 15227903 IC50 > 50000 nM T30081 CYQ94X 15227904 IC50 > 50000 nM T30081 C5KD4V 15227905 IC50 > 50000 nM T30081 CU8B2A 15227906 IC50 > 50000 nM T30081 CWX5O0 15227907 IC50 > 50000 nM T30081 CT0CV1 15227908 IC50 > 50000 nM T30081 C4MUA1 22489180 IC50 > 1000000 nM T30081 CM91RP 24750302 IC50 > 500000 nM T30081 C07PEZ 24750303 IC50 > 500000 nM T30081 CTO90W 24750304 IC50 > 500000 nM T30081 CW2HP5 24750413 IC50 > 500000 nM T30081 C6ZE3D 44269001 Ki = 2000 nM T30081 C0R2AF 44286728 IC50 = 25000 nM T30081 CH4E8O 44286741 IC50 > 50000 nM T30081 CXTL42 44286784 IC50 > 50000 nM T30081 C9TFB7 44286896 Ki = 4300 nM T30081 CU5C7P 44333373 IC50 = 33000 nM T30081 C6CBN2 44333378 IC50 = 28000 nM T30081 C0EU3K 44333390 IC50 = 3500 nM T30081 CGYW24 44333414 IC50 = 180000 nM T30081 C76KRP 44333420 IC50 = 23000 nM T30081 C09IHV 44333437 IC50 = 491000 nM T30081 CGK2H1 44333745 IC50 = 27000 nM T30081 C12KRO 44333760 IC50 = 4100 nM T30081 CB5C8I 44355754 IC50 = 11000 nM T30081 C4G8PD 44355755 IC50 = 28000 nM T30081 CVH87D 44355905 IC50 = 4600 nM T30081 CR6Y8V 44355914 IC50 = 20000 nM T30081 CP9QL3 44355988 IC50 = 17000 nM T30081 C6ZO2D 44356613 IC50 = 19000 nM T30081 C17QOA 44420577 IC50 > 500000 nM T30081 C9HVL3 44420578 IC50 > 500000 nM T30081 CHP3U9 44420579 IC50 > 500000 nM T30081 CIQ47X 44420582 IC50 > 500000 nM T30081 CQY8X5 44437450 IC50 > 1000000 nM T30081 C5H7LS 44437451 IC50 > 1000000 nM T30081 CD0AN5 44437452 IC50 > 500000 nM T30081 C4YH3T 44437453 IC50 > 1000000 nM T30081 C2QO0P 44437477 IC50 > 500000 nM T30081 C9OE0G 44437478 IC50 > 500000 nM T30081 CO0N8X 44437480 IC50 > 1000000 nM T30081 C4V2AD 44560487 IC50 = 13000 nM T30081 CPM1F3 44560491 IC50 = 405000 nM T30081 C2XN5Q 44560560 IC50 = 10000 nM T30081 C3BJE2 46197226 IC50 > 500000 nM T30081 C8WR4I 46197456 IC50 > 500000 nM T30081 C2Y0QN 46197457 IC50 > 500000 nM T30081 CPA6D7 46700799 IC50 = 366000 nM T30081 CWJY16 46874452 IC50 > 500000 nM T30081 C1PCR5 46884564 IC50 = 71000 nM T30081 C4NK8W 46884565 IC50 = 75000 nM T30081 C48RWL 46884566 IC50 >= 500000 nM T30081 CN9RI6 46884567 IC50 = 109000 nM T30081 C8DP0M 46885250 IC50 = 316000 nM T30081 CQWV32 46885301 IC50 = 318000 nM T30081 CG74UX 46885302 IC50 = 177000 nM T30081 C9V5IT 46888106 IC50 = 105000 nM T30081 CB6PI7 46888107 IC50 = 311000 nM T30081 CB3V5I 46888108 IC50 = 114000 nM T30081 C9DI3F 46888151 IC50 = 86000 nM T30081 C9MZK2 46888152 IC50 = 60000 nM T30081 CUR4G7 46913823 IC50 = 200 ug.mL-1 T30081 CSQL06 54768280 IC50 = 200 ug.mL-1 T30081 CB9DU0 54768281 IC50 = 200 ug.mL-1 T30081 CUN04G 54768283 IC50 = 200 ug.mL-1 T30081 C2P3CT 90663608 IC50 > 1000000 nM T30081 C7MA3K 135398592 IC50 = 115000 nM T30081 C6Z4QV 135425312 Ki = 25000 nM T30081 C63BVC 135433410 Ki = 2060 nM T30081 CV0HE2 135499520 IC50 > 500000 nM T30081 C4K1FL 136118006 IC50 > 500000 nM T30081 CQGF80 136118007 IC50 > 500000 nM T30081 CR37CF 136118008 IC50 > 500000 nM T30081 D01GLG 5789 IC50 = 26 nM T30081 D0C7YS 160155 Ki = 20000 nM T30081 D0G5VO 135415618 Ki = 50 nM T30081 D0I6UV 6477686 IC50 = 180 nM T30081 D0M4MA 6035 Ki = 5060 nM T30081 D0O7GD 452142 IC50 >= 500000 nM T55781 D03ZBT 11626560 IC50 > 100 nM T55781 D0C4RB 36314 IC50 = 4900 nM T55781 D0W5HK 216239 IC50 = 1370 nM T55781 D00DRL 44137946 IC50 = 24 nM T55781 D03LWG 53235510 IC50 > 10000 nM T55781 D05PZB 135398495 IC50 = 1 nM T55781 D06DMQ 59472121 Ki = 30 nM T55781 D0E3TC 44259 IC50 = 11.6 nM T55781 D0O6WV 24794418 IC50 = 14 nM T55781 D03BNU 59604787 IC50 > 10000 nM T55781 D03RHV 72793043 IC50 = 600 nM T55781 D08OEW 72792975 IC50 = 72 nM T55781 D0M9TR 72793042 IC50 = 1130 nM T55781 CGAN35 2856 IC50 = 11000 nM T55781 CWQ7U1 696836 IC50 = 2060 nM T55781 C1C5EJ 784137 IC50 > 30000 nM T55781 CACS26 11561968 Ki > 2000 nM T55781 CU0E8O 11690457 Ki > 2000 nM T55781 CF57GK 46215462 IC50 = 15 nM T55781 CG6KA7 50945534 IC50 > 30000 nM T55781 CJ98GR 50947631 IC50 = 2250 nM T55781 C1SA2T 52109814 IC50 = 3560 nM T55781 CV8U6Y 52110137 IC50 = 680 nM T55781 CXSE16 52111270 IC50 = 4170 nM T55781 C3RC8Q 52111275 IC50 = 1240 nM T55781 CSF0Q5 52111278 IC50 = 1080 nM T55781 CUPV64 52111292 IC50 = 2900 nM T55781 C3V5XE 53355503 IC50 = 2.9 nM T55781 CC62KV 54915268 IC50 = 3000 nM T55781 CBOD63 56835089 IC50 = 2440 nM T55781 CD6Y9Z 57395116 IC50 = 2340 nM T55781 C8W6IG 57395117 IC50 = 970 nM T55781 CG7S0D 57396882 IC50 = 6930 nM T55781 C1MR8Q 60097495 IC50 > 1000 nM T55781 C10AMI 66553589 IC50 > 10000 nM T55781 CV63UL 67240318 IC50 > 10000 nM T55781 CJLT43 67471113 IC50 = 56 nM T55781 CXR9Y0 68212353 IC50 = 120 nM T55781 CEH69L 68212361 IC50 = 25 nM T55781 C4V3DJ 68212395 IC50 = 56 nM T55781 CPZ8D7 68212421 IC50 = 140 nM T55781 CBUE63 68212479 IC50 = 1400 nM T55781 CR0B8N 68212480 IC50 = 1.8 nM T55781 CZJ83X 68212482 IC50 = 0.25 nM T55781 C1QXE9 68212489 IC50 = 62 nM T55781 C5H8DO 68212494 IC50 = 4500 nM T55781 C2WDO9 68212498 IC50 = 74 nM T55781 C7PT2D 68212505 IC50 = 0.76 nM T55781 CKPF54 68212509 IC50 = 0.15 nM T55781 C40GFP 68212528 IC50 = 7000 nM T55781 CJY4P6 68212724 IC50 = 18 nM T55781 C2ZCD6 68212733 IC50 = 10 nM T55781 C4ARE2 68212746 IC50 = 8.2 nM T55781 CTM2R4 68212750 IC50 = 530 nM T55781 C5MG7K 68212755 IC50 = 13 nM T55781 COV36W 68212757 IC50 = 5.8 nM T55781 C51DUT 68212759 IC50 = 13 nM T55781 CL95KS 68212760 IC50 = 200 nM T55781 CQD3H2 68212763 IC50 = 400 nM T55781 C6GU4S 68212779 IC50 = 2400 nM T55781 CG5VP7 68212780 IC50 = 860 nM T55781 CJR90K 68212791 IC50 = 10 nM T55781 CS5C0R 68212798 Ki = 0.33 nM T55781 C2B8DE 70681768 IC50 = 9600 nM T55781 CQAU72 70681769 IC50 = 170 nM T55781 CG80HU 70681780 Ki = 2 nM T55781 C8JYH4 70686029 IC50 = 2800 nM T55781 C7LVS2 70692345 IC50 = 14 nM T55781 CWP13X 70695379 IC50 = 2400 nM T55781 CM0D3O 70696465 IC50 = 28000 nM T55781 CTB5O3 70696471 IC50 = 64 nM T55781 C5Q3YE 70697396 IC50 = 2200 nM T55781 CH0B8N 70789756 IC50 = 4680 nM T55781 CA3O6K 71552696 IC50 = 126 nM T55781 C1NPL0 71552941 IC50 = 1920 nM T55781 CA4PS8 71552942 IC50 = 775 nM T55781 C4Q2HC 71721525 IC50 = 4.3 nM T55781 CQ3JN8 71819732 IC50 = 17 nM T55781 C9NVM8 72192165 IC50 = 5.2 nM T55781 C7A8XR 72547635 IC50 = 150 nM T55781 CUPN10 72547636 IC50 = 37 nM T55781 C5MI7D 72547637 IC50 = 11 nM T55781 CD93WQ 72547638 IC50 = 24 nM T55781 C49RTS 72547864 IC50 = 120 nM T55781 C45UFT 72547868 IC50 = 180 nM T55781 CM23ZS 72548104 IC50 = 47 nM T55781 CO7MN3 72548105 IC50 > 30000 nM T55781 CH05EK 72551069 IC50 = 23 nM T55781 C07THM 72551070 IC50 = 40 nM T55781 CVNK29 72551073 IC50 = 2.1 nM T55781 CO3UW2 72551074 IC50 = 9 nM T55781 CP09RS 72792559 IC50 > 30000 nM T55781 C3PTC7 72792560 IC50 = 12 nM T55781 C12IMZ 72792561 IC50 = 18 nM T55781 C2E0RN 72792562 IC50 = 1.1 nM T55781 CZXU21 72792563 IC50 = 1.7 nM T55781 CD7UM4 72792564 IC50 = 0.7 nM T55781 C38OCL 72792627 IC50 = 0.69 nM T55781 C39PHS 72792906 IC50 = 3.4 nM T55781 C6HYA4 72792907 IC50 = 0.69 nM T55781 C16ETP 72792908 IC50 = 1.3 nM T55781 CNSX89 72792909 IC50 = 0.81 nM T55781 C7HXN3 72792910 IC50 = 1250 nM T55781 CGP01I 72792971 IC50 = 1.8 nM T55781 CXNF57 72792972 IC50 = 4.5 nM T55781 CGDL83 72792973 IC50 = 18 nM T55781 CJGF34 72792974 IC50 = 34 nM T55781 C4N9TK 72792977 IC50 = 200 nM T55781 C5B9CI 72793044 IC50 > 30000 nM T55781 C86UHM 72793045 IC50 = 2700 nM T55781 C75QHA 72793046 IC50 = 540 nM T55781 C1MPN7 72793047 IC50 = 170 nM T55781 CRJ81Y 72793048 IC50 = 50 nM T55781 CL9EA5 72793105 IC50 = 19 nM T55781 CVT7A9 72793106 IC50 = 44 nM T55781 C39VXU 72793107 IC50 = 380 nM T55781 C43SNK 72793108 IC50 = 16500 nM T55781 C9XAE8 72793109 IC50 = 83 nM T55781 CZA34R 72793110 IC50 = 110 nM T55781 CU9R4X 72793111 IC50 = 14 nM T55781 CD2K0R 72793177 IC50 = 320 nM T55781 CP26TN 72793178 IC50 = 220 nM T55781 CKV95R 72793179 IC50 = 44 nM T55781 CH80BD 72793182 IC50 = 12600 nM T55781 CAJ65L 72793183 IC50 > 30000 nM T55781 CVR1I4 72793252 IC50 = 67 nM T55781 CJWB46 72793253 IC50 = 5900 nM T55781 CMIH15 72793254 IC50 = 2500 nM T55781 C30IXP 72793255 IC50 = 8.4 nM T55781 C6YFO5 72793256 IC50 = 4.1 nM T55781 CJG79M 72793257 IC50 = 13 nM T55781 CK6U5Z 72793332 IC50 = 8 nM T55781 CI6JX5 72793333 IC50 = 230 nM T55781 CA4ET8 72793334 IC50 = 15 nM T55781 C6JW5N 72793335 IC50 = 29 nM T55781 CROW51 72793336 IC50 = 39 nM T55781 C65KJA 72793337 IC50 = 14 nM T55781 C7IA8R 72793397 IC50 = 6.7 nM T55781 CD85ZE 72793399 IC50 = 6.3 nM T55781 CI4E7H 72793400 IC50 = 14 nM T55781 C02GET 72793401 IC50 = 590 nM T55781 C9WYE4 72793466 IC50 = 37 nM T55781 C37FKG 72793468 IC50 = 62 nM T55781 COU2I8 72793469 IC50 = 1000 nM T55781 C49MHY 72793532 IC50 = 110 nM T55781 C3K2BV 72793533 IC50 = 620 nM T55781 C5UH4O 72793534 IC50 = 170 nM T55781 C2Z6FI 72793535 IC50 = 9900 nM T55781 CLTB82 72793536 IC50 = 2400 nM T55781 CQ7KX1 72793601 IC50 = 18 nM T55781 CW0PY4 72793602 IC50 = 570 nM T55781 CKB3O6 72793603 IC50 = 950 nM T55781 CI9L8K 72793604 IC50 = 15200 nM T55781 CMD9F8 72793605 IC50 = 6.3 nM T55781 CE60AT 72793606 IC50 = 2.8 nM T55781 C75UBS 72793607 IC50 = 3.9 nM T55781 C51VIE 72793608 IC50 = 27 nM T55781 COL6Y5 72793609 IC50 = 7.3 nM T55781 CJ9C7M 72793610 IC50 = 86 nM T55781 CGCL01 72793611 IC50 = 59 nM T55781 CZ5QY9 72793612 IC50 > 30000 nM T55781 CJ87CG 73211763 IC50 = 1.7 nM T55781 C1V3NZ 73425588 IC50 = 0.74 nM T55781 CQ4ZH2 74538669 IC50 = 4.4 nM T55781 CG7VE4 76309971 IC50 = 140 nM T55781 C17BGH 76328134 IC50 = 160 nM T55781 CH8W7D 77461036 IC50 > 1000 nM T55781 CHIZ70 89495685 IC50 = 1.3 nM T55781 CS6IA4 89495748 IC50 = 1.6 nM T55781 CW1OS0 89495775 IC50 = 0.57 nM T55781 C61JAN 91966173 IC50 = 7840 nM T55781 CQVL13 91966182 IC50 = 3430 nM T55781 CL2DH6 118433464 IC50 = 3.2 nM T55781 C01OAD 118433470 IC50 = 4.9 nM T55781 C9ENZ0 118433703 IC50 = 5.2 nM T55781 CQU1R4 118443520 IC50 = 22 nM T55781 C8OSQ4 118443521 IC50 = 3.5 nM T55781 CAM76F 118443524 IC50 = 3.6 nM T55781 C3DEP2 118443546 IC50 = 4.3 nM T55781 CGO6B1 118443548 IC50 = 1068 nM T55781 CADG96 118443549 IC50 = 5.2 nM T55781 CM92EG 118443553 IC50 = 19 nM T55781 CVWR20 118443556 IC50 = 20 nM T55781 CC9FK0 118443560 IC50 = 2.6 nM T55781 CRZ68N 118443583 IC50 = 2.5 nM T55781 C9I5MC 118443585 IC50 = 4.9 nM T55781 CE42TF 118443586 IC50 = 72 nM T55781 C5YJT1 118443594 IC50 = 2 nM T55781 CL0YO5 118443595 Ki = 0.43 nM T55781 CG3K5V 118443597 IC50 = 3.5 nM T55781 C12WAU 118446433 IC50 = 78 nM T55781 CFBY13 118446434 IC50 = 3.5 nM T55781 CY6C1E 122179442 IC50 > 10000 nM T55781 C08KEM 122179540 IC50 = 5400 nM T55781 CG0RP7 122179547 IC50 = 4700 nM T55781 C1A0SQ 122179548 IC50 = 5100 nM T55781 C8KXV1 127025843 IC50 > 1000 nM T55781 CB5JD0 127043185 IC50 = 10200 nM T55781 CRC8Y3 127043566 IC50 > 30000 nM T55781 CV7L1K 127043900 IC50 = 1840 nM T55781 C34VIW 127045062 IC50 > 30000 nM T55781 CS9H0C 127045063 IC50 = 7270 nM T55781 C2QDF3 127045215 IC50 = 1720 nM T55781 C4KH2E 127045219 IC50 > 30000 nM T55781 CK36LR 127045379 IC50 > 30000 nM T55781 CWJ1H6 127045411 IC50 = 1140 nM T55781 C0Q7TL 127045560 IC50 = 2010 nM T55781 C9LP2C 127045567 IC50 > 30000 nM T55781 C8ERJ7 127045762 IC50 > 1000 nM T55781 C7JC5K 134132904 IC50 = 1.8 nM T55781 C5DSV1 134134351 IC50 = 54 nM T55781 CYB46P 134135659 IC50 = 150 nM T55781 CDH31O 134136945 EC50 = 34 nM T55781 C46XTD 134138113 IC50 = 86 nM T55781 CK75ZI 134138785 IC50 = 13 nM T55781 CCE1O4 134138988 IC50 = 3 nM T55781 C9V4CG 134140406 EC50 = 150 nM T55781 C5C4TS 134141052 IC50 = 94 nM T55781 CWI41J 134141468 EC50 = 490 nM T55781 CYM06R 134142159 IC50 = 160 nM T55781 CZB68J 134142873 EC50 = 210 nM T55781 CX03CP 134143856 IC50 = 140 nM T55781 C5C2TA 134144975 IC50 = 4 nM T55781 CE12IN 134145489 IC50 = 170 nM T55781 CM4U6L 134147181 IC50 = 9.6 nM T55781 CBES34 134147807 IC50 = 4.1 nM T55781 C60FLZ 134148014 EC50 = 150 nM T55781 CDUX09 134148124 IC50 = 65 nM T55781 CGIT02 134149104 IC50 = 4.1 nM T55781 C4CA2M 134149641 IC50 = 17 nM T55781 C36GLZ 134150279 EC50 = 160 nM T55781 CZ42MI 134150952 IC50 = 11 nM T55781 C39AMZ 134151100 EC50 = 72 nM T55781 C10BFN 134151512 IC50 = 30 nM T55781 C8M3RH 134152780 IC50 = 5 nM T55781 C5PV8R 134153049 IC50 = 3.9 nM T55781 C4M7XF 134153576 IC50 = 80 nM T55781 C4AR9L 134153778 EC50 = 690 nM T55781 C6GC3U 134154700 IC50 = 8.9 nM T55781 C20PJY 134156194 IC50 = 5.6 nM T55781 CHN5R6 134156911 IC50 = 16 nM T55781 C70ZRI 134157187 IC50 = 4.9 nM T55781 CXC69T 137321158 IC50 = 29 nM T55781 C25ERN 137631967 IC50 = 4.4 nM T55781 C06JRX 137637094 IC50 = 36.9 nM T55781 C7TG3J 137641313 IC50 = 7585.78 nM T55781 C1DK0P 137651391 IC50 = 7.1 nM T55781 CV5H3Z 137657932 IC50 = 30.9 nM T55781 CE84NX 144944001 IC50 = 24 nM T55781 C65YWX 145964882 IC50 = 2500 nM T55781 CHC3T0 145965031 IC50 > 10000 nM T55781 CP92ZF 145965329 IC50 = 640 nM T55781 C9HXI4 145966620 IC50 = 2300 nM T55781 CQE9M5 145966810 IC50 = 480 nM T55781 C1EH6C 145967078 IC50 = 8700 nM T55781 CWJ12M 145969155 IC50 = 92 nM T55781 CGW5S1 145969844 IC50 = 2000 nM T55781 CB8R3A 145970271 IC50 > 10000 nM T55781 C40VIL 145972979 IC50 = 6200 nM T55781 CQBY19 145974023 IC50 > 10000 nM T55781 C4X7CT 145977420 IC50 = 5400 nM T55781 CLA57T 145978300 IC50 = 8900 nM T55781 C6KDQ5 145979093 IC50 = 22 nM T55781 CV7QY8 145981517 IC50 = 3.1 nM T55781 CG0R3A 145984368 IC50 = 90 nM T55781 CV78XO 145985621 IC50 = 61 nM T55781 CX5MB2 145986730 IC50 = 13 nM T55781 C1V6RA 145988134 IC50 > 100000 nM T55781 CD98JK 145989189 IC50 = 13 nM T55781 CWH69B 145989428 IC50 = 2.2 nM T55781 CZCS58 145989494 IC50 = 1.2 nM T55781 C0PHA7 145990595 IC50 = 40 nM T55781 CN6T4K 145991513 IC50 = 9 nM T55781 CMBH76 145991936 IC50 = 1.3 nM T55781 C0SO4N 145993259 IC50 = 4.9 nM T55781 CI7F4G 145994227 IC50 = 4.1 nM T55781 CL4B2M 155512535 IC50 = 2630 nM T55781 C81YCJ 155513061 IC50 = 3120 nM T55781 CTSM92 155538441 IC50 = 25 nM T55781 CC5F3I 155562216 IC50 = 3950 nM T55781 C40IYS 155562258 IC50 = 4.2 nM T55781 D0N4LR 53469448 IC50 = 474 nM T55781 D0Q0YV 24944925 IC50 = 6456.54 nM T99455 D00STL 644241 IC50 = 12.7 nM T99455 D0AZ3C 5291 IC50 = 14 nM T99455 D0E6XR 3062316 EC50 = 0.04 nM T99455 D0H0EQ 24826799 EC50 = 0.05 nM T99455 D0OB0F 5328940 IC50 = 20 nM T99455 D0R0MW 5329102 EC50 > 1000 nM T99455 D02LJW 23635314 IC50 = 100 nM T99455 D02XNW 5494449 IC50 = 50.12 nM T99455 D06JHV 46848036 IC50 = 6.2 nM T99455 D0E3TC 44259 IC50 = 121.8 nM T99455 D0U3EP 445154 IC50 = 28000 nM T99455 D05HDJ 49782106 EC50 = 7150 nM T99455 D0EF5T 44129660 EC50 = 430 nM T99455 D0JY1I 42613483 IC50 = 2700 nM T99455 D0L7XM 42628828 EC50 = 40 nM T99455 D0OE4F 4369496 IC50 = 100 nM T99455 D0ZH4I 76071870 IC50 > 10000 nM T99455 D01EFO 9864718 IC50 = 398.11 nM T99455 C6SB2N 123596 EC50 = 90 nM T99455 CV5MS2 2475277 EC50 = 1300 nM T99455 CCPF82 5312285 EC50 = 720 nM T99455 CZR3M4 9799152 IC50 = 100000 nM T99455 CY3MK1 9807952 IC50 = 3.981 nM T99455 CI3O6X 9814609 IC50 = 61659.5 nM T99455 CX9DG5 9822042 IC50 = 199.53 nM T99455 CSH0A9 9847014 IC50 = 346.74 nM T99455 C3UQL7 9860872 IC50 = 33884.42 nM T99455 CC90FJ 9869737 IC50 = 512 nM T99455 CIZ13L 9943193 IC50 = 602.56 nM T99455 CUKH27 9943194 IC50 = 707.95 nM T99455 CU78NO 9947433 IC50 = 151.36 nM T99455 CYT7R9 9953676 IC50 = 794.33 nM T99455 CJ40GO 9965429 IC50 = 1513.56 nM T99455 CTE3K0 9982070 IC50 = 3162.28 nM T99455 CP23QA 10007129 IC50 = 10 nM T99455 CLI9A3 10029363 IC50 = 63.1 nM T99455 C0G5DK 10039959 IC50 = 7943.28 nM T99455 CT9F2H 10053560 IC50 = 5.012 nM T99455 C8EW6P 10095381 IC50 = 2187.76 nM T99455 C3P8WK 10110378 IC50 = 1000 nM T99455 C63CFD 10111108 IC50 = 1288.25 nM T99455 CL42XS 10136330 IC50 = 794.33 nM T99455 CUW34X 10157645 IC50 = 1905.46 nM T99455 COC30E 10181160 IC50 = 199.53 nM T99455 CN51JQ 10292737 IC50 = 446.68 nM T99455 CG2L4Z 10343860 IC50 = 602.56 nM T99455 CYW13A 10348904 IC50 = 10 nM T99455 C7TJ9U 10483163 IC50 = 7.079 nM T99455 CS0DE8 10493971 IC50 > 3000 nM T99455 C78FPR 10501266 IC50 = 371.54 nM T99455 CU6G5Y 10708835 IC50 = 1202.26 nM T99455 CO61VZ 11161166 IC50 = 24000 nM T99455 C94MLD 11165739 EC50 = 390 nM T99455 C2KT9E 11168002 IC50 = 4.074 nM T99455 C89EZO 11180525 IC50 = 16.98 nM T99455 C3FL9M 11199480 IC50 > 100000 nM T99455 CJTP13 11280103 IC50 = 3801.89 nM T99455 CPW2Y8 11326963 EC50 = 4470 nM T99455 C1DF5Z 11336923 EC50 = 330 nM T99455 CKY3E2 11338122 IC50 = 199.53 nM T99455 CH4O8K 11347791 EC50 = 1660 nM T99455 C4RLW0 11368874 IC50 = 26000 nM T99455 C3OCV2 11371778 IC50 = 1000 nM T99455 CHJV86 11381980 EC50 = 470 nM T99455 C14XYD 11385486 IC50 > 10000 nM T99455 C3O0WI 11438191 IC50 = 5128.61 nM T99455 C3EXM4 11440028 IC50 = 398.11 nM T99455 C2E0GS 11461932 EC50 = 1800 nM T99455 C7I6AG 11474111 IC50 = 501.19 nM T99455 C0YH2X 11478363 IC50 = 1.25 nM T99455 CMW72Q 11488124 IC50 = 724.44 nM T99455 C57TKI 11565665 IC50 = 18000 nM T99455 C43JZU 11604436 IC50 = 3800 nM T99455 CGU7N0 11604739 IC50 = 12900 nM T99455 CLJ81E 11630507 IC50 = 20000 nM T99455 C6SGF3 11644985 IC50 = 16000 nM T99455 CJK78Z 11652152 IC50 = 8000 nM T99455 CAJS96 11662893 IC50 = 14600 nM T99455 CH3S9K 11666294 IC50 = 20000 nM T99455 C95EPO 11666668 IC50 = 35000 nM T99455 CKAH36 11669784 IC50 = 9500 nM T99455 CJ89UZ 11687939 IC50 > 100000 nM T99455 C7RDH3 11709536 IC50 > 100000 nM T99455 CFJ4I7 11723151 IC50 = 3311.31 nM T99455 C7C2FM 11737638 IC50 = 1513.56 nM T99455 CVFS29 11751305 IC50 = 64.57 nM T99455 CPJ7C9 11774222 EC50 = 580 nM T99455 CUDO23 11994441 IC50 = 25.12 nM T99455 C02DIH 14347011 IC50 = 1819.7 nM T99455 CZB2V0 16750146 IC50 = 20.89 nM T99455 C6XC2W 23145852 IC50 = 10.96 nM T99455 CUVB29 23145858 IC50 = 3.981 nM T99455 CO0T3M 24825778 IC50 = 750 nM T99455 CIFO50 24897305 IC50 = 11000 nM T99455 CYXC26 24958918 IC50 = 10000 nM T99455 CVUK27 24958920 IC50 = 2500 nM T99455 C35LZO 24959284 IC50 = 2500 nM T99455 CIZQ04 24959285 IC50 = 15000 nM T99455 C47ING 24959648 IC50 = 10000 nM T99455 C4V9GI 24960018 IC50 = 500 nM T99455 CWLR85 24960379 IC50 = 10000 nM T99455 CHC6A5 25017304 IC50 = 1378 nM T99455 C38YMD 25017555 IC50 = 7083 nM T99455 CDHM05 25017557 IC50 = 739.5 nM T99455 CFU60Y 25235817 IC50 = 436 nM T99455 C8B6TY 42628503 EC50 < 500 nM T99455 C15OSL 42633116 EC50 = 250 nM T99455 CO1I2D 42633117 EC50 = 1200 nM T99455 CO7YL0 42633119 EC50 > 10000 nM T99455 CWF2S8 42633305 EC50 = 160 nM T99455 CKCO80 42633306 EC50 = 400 nM T99455 CCI8P7 42633666 EC50 = 1320 nM T99455 CSH3I9 42633667 EC50 = 2200 nM T99455 CPNK96 42633668 EC50 = 4340 nM T99455 CL04QK 42633670 EC50 > 10000 nM T99455 C7DA0B 42633859 EC50 = 9680 nM T99455 CLM7B9 42634040 EC50 = 490 nM T99455 C6DK1W 42634389 EC50 > 10000 nM T99455 C87GKI 42634390 EC50 = 918 nM T99455 CK15FQ 42634392 EC50 = 406 nM T99455 CCN5O4 42634553 EC50 = 1340 nM T99455 C2H1SJ 42634556 EC50 = 48 nM T99455 C1M8SR 42634557 EC50 = 1960 nM T99455 C48YFI 42634730 EC50 = 5600 nM T99455 C8L5RN 42635093 EC50 = 150 nM T99455 CQ9F8I 42635272 EC50 = 120 nM T99455 CG2P1M 42635644 EC50 = 1230 nM T99455 C4JRG0 42635811 EC50 = 140 nM T99455 CCOV80 42635815 EC50 = 100 nM T99455 C7K9YE 44194683 EC50 = 420 nM T99455 C9G6QE 44194684 EC50 = 340 nM T99455 CBP7D2 44194685 EC50 = 240 nM T99455 CBD90A 44194780 EC50 = 920 nM T99455 COK3J5 44194781 EC50 = 970 nM T99455 C7XOD2 44194782 EC50 = 1150 nM T99455 C4T0HN 44194783 EC50 = 1270 nM T99455 C63UIZ 44194784 EC50 = 1240 nM T99455 CMRX16 44273620 IC50 = 5754.4 nM T99455 CCH89M 44300026 IC50 = 1995.26 nM T99455 CH4ND7 44340691 IC50 = 9772.37 nM T99455 CK2CU3 44340703 IC50 = 17378.01 nM T99455 CY0XF5 44340726 IC50 = 67608.3 nM T99455 C2F7SL 44395745 IC50 = 10000 nM T99455 C0TED6 44395746 IC50 = 5011.87 nM T99455 CZR42M 44395763 IC50 = 575.44 nM T99455 CJ0Z5K 44395813 IC50 = 8912.51 nM T99455 CU9XQ0 44395880 IC50 = 10000 nM T99455 CYF8U6 44395904 IC50 = 1000 nM T99455 C5DR6W 44395926 IC50 = 10000 nM T99455 C4R8EB 44410932 IC50 = 23000 nM T99455 CI82UE 45270897 IC50 > 10000 nM T99455 C4UM6Y 45273507 IC50 > 10000 nM T99455 CR4A6B 46703970 EC50 > 10000 nM T99455 CH9AW2 46865999 IC50 = 500 nM T99455 C4FX6S 46866098 IC50 = 500 nM T99455 CK6UL0 46866099 IC50 = 200 nM T99455 C67UEP 46881960 IC50 = 8 nM T99455 C71XDW 49780994 EC50 = 330 nM T99455 CEAH78 49780998 EC50 = 5000 nM T99455 CHS50Y 49780999 EC50 = 2920 nM T99455 C9WOE2 49781000 EC50 = 480 nM T99455 CGV34K 49781215 EC50 = 90 nM T99455 C84ZOI 49781216 EC50 = 360 nM T99455 C4K9DH 49781217 EC50 = 810 nM T99455 C34JPY 49781218 EC50 = 400 nM T99455 C7YET3 49781219 EC50 = 290 nM T99455 C48NTZ 49781220 EC50 = 170 nM T99455 C7QON3 49781221 EC50 > 10000 nM T99455 CHUG72 49781431 EC50 > 10000 nM T99455 CQ43VM 49781432 EC50 > 10000 nM T99455 CDU34O 49781433 EC50 > 10000 nM T99455 CSE62H 49781434 EC50 > 10000 nM T99455 CL51PM 49781435 EC50 > 10000 nM T99455 CE1N9P 49781436 EC50 > 10000 nM T99455 CF4TU7 49781437 EC50 > 10000 nM T99455 CH4MI1 49781662 EC50 > 10000 nM T99455 CQOW70 49781663 EC50 > 10000 nM T99455 C46TMR 49781664 EC50 > 10000 nM T99455 CG2I3L 49781665 EC50 > 10000 nM T99455 COW0H6 49781667 EC50 > 10000 nM T99455 CBH02L 49781668 EC50 = 1440 nM T99455 C6-DEC-09 49781877 EC50 > 10000 nM T99455 CGI64U 49781878 EC50 = 6890 nM T99455 C38FVM 49781879 EC50 = 380 nM T99455 CVT73X 49781880 EC50 = 760 nM T99455 C7X9UG 49781881 EC50 = 300 nM T99455 C5I3OF 49781882 EC50 = 270 nM T99455 C1T6CN 49782104 EC50 = 400 nM T99455 C6WOK4 49782105 EC50 = 350 nM T99455 CKQC50 49782107 EC50 = 6890 nM T99455 CWHY47 49782108 EC50 = 690 nM T99455 CGC82O 49782109 EC50 = 2960 nM T99455 C80XEK 49782334 EC50 = 6920 nM T99455 C2BNW5 49782337 EC50 = 160 nM T99455 C1EA9K 49782338 EC50 = 1700 nM T99455 C2Y6QS 50938552 IC50 > 10000 nM T99455 CS3LT9 51030149 IC50 = 671 nM T99455 C1XRG0 51030150 IC50 = 507 nM T99455 C3PDJ8 51030250 IC50 = 774 nM T99455 CAQ4V6 51030532 IC50 = 480 nM T99455 CX47EM 51030534 IC50 = 1300 nM T99455 CSZ36G 51030713 IC50 = 177 nM T99455 CA6U5X 51030714 IC50 = 491 nM T99455 C9NYP4 51036677 IC50 > 10000 nM T99455 C4WRY3 51037112 IC50 > 10000 nM T99455 CNWO03 51037408 IC50 = 5 nM T99455 CLO1I6 51037410 IC50 = 6 nM T99455 CZ2H3T 51037608 IC50 = 19 nM T99455 CK8J5T 51037609 IC50 = 904 nM T99455 CYO9W0 51037823 IC50 = 458 nM T99455 CF7HX6 51037824 IC50 = 161 nM T99455 CMX3I7 51037825 IC50 = 19 nM T99455 CRI28Z 51037948 IC50 > 10000 nM T99455 C4XT7P 51038497 IC50 = 24 nM T99455 CKB79R 51038498 IC50 = 125 nM T99455 C75JSI 51038499 IC50 = 7 nM T99455 C6PG5F 51351510 IC50 = 20.1 nM T99455 CHAV48 52940594 IC50 = 2500 nM T99455 CAK80G 52940928 IC50 = 2500 nM T99455 C02ALP 52940992 IC50 > 20000 nM T99455 CSM30J 52941799 IC50 = 2500 nM T99455 CFY5K7 52941942 IC50 = 10000 nM T99455 CPU53W 52941997 IC50 = 2500 nM T99455 C1LN4J 52942048 IC50 = 500 nM T99455 C69VKZ 52942052 IC50 = 2500 nM T99455 C0QFI8 52942203 IC50 > 20000 nM T99455 C7D5FE 52942236 IC50 > 20000 nM T99455 C0S7OM 52943049 IC50 = 2500 nM T99455 CQZ98C 52943259 IC50 = 2500 nM T99455 CZ3X7O 52943392 IC50 > 20000 nM T99455 C9L3HD 52943395 IC50 = 20000 nM T99455 CCBA25 52944595 IC50 > 20000 nM T99455 C1XN6P 52944599 IC50 > 20000 nM T99455 C1H8GZ 52944627 IC50 > 20000 nM T99455 C90JQR 52945824 IC50 > 20000 nM T99455 CPVD21 52945847 IC50 > 20000 nM T99455 C62EXZ 52946812 IC50 = 10000 nM T99455 C3WI7B 52947902 IC50 = 2500 nM T99455 CK08IW 52948022 IC50 = 2500 nM T99455 CJ1XR3 52948871 EC50 > 10000 nM T99455 C4Q6XB 52949498 IC50 > 20000 nM T99455 CCXY64 54581006 IC50 = 5510 nM T99455 C36DEH 54582045 IC50 = 277 nM T99455 CPI87W 54583990 IC50 > 2000 nM T99455 CIE67G 54585892 IC50 = 3780 nM T99455 CAIO65 68796885 EC50 = 0.04 nM T99455 C91HPI 71300299 IC50 > 5000 nM T99455 CC98EU 71449991 IC50 = 2.67 nM T99455 CV21PC 71449992 IC50 = 5.96 nM T99455 CG59TB 71449993 IC50 = 0.45 nM T99455 C23ETA 71450038 IC50 = 1.66 nM T99455 C3B7IP 71450039 IC50 = 0.36 nM T99455 C0XL6Z 71451816 IC50 = 2.25 nM T99455 CQM05U 71451817 IC50 = 0.6 nM T99455 CVE9P2 71451818 IC50 = 0.52 nM T99455 C30FHU 71453635 IC50 = 0.54 nM T99455 CR7DI8 71453636 IC50 = 1.01 nM T99455 C8K6BL 71453637 IC50 = 19.1 nM T99455 C12IUO 71453638 IC50 = 0.52 nM T99455 CIEK84 71453639 IC50 = 0.72 nM T99455 C0FTX4 71453675 IC50 = 0.33 nM T99455 CK7V6O 71453676 IC50 = 0.42 nM T99455 CU42QX 71455363 IC50 = 0.52 nM T99455 C4X9GT 71455364 IC50 = 0.78 nM T99455 CVY26H 71455365 IC50 = 1.18 nM T99455 C3X1OP 71455406 IC50 = 0.52 nM T99455 COUR46 71455407 IC50 = 1.03 nM T99455 C8IV0R 71455408 IC50 = 1.01 nM T99455 CY2G7S 71457180 IC50 = 0.7 nM T99455 CXA9W8 71457181 IC50 = 0.98 nM T99455 CCT0X3 71459003 IC50 = 17.8 nM T99455 C01XBA 71459004 IC50 = 2.56 nM T99455 C0WF3X 71459043 IC50 = 1.94 nM T99455 CJ3PO5 71459044 IC50 = 15 nM T99455 CW0X4B 71460798 IC50 = 3.44 nM T99455 CE84WT 71460799 IC50 = 12.8 nM T99455 CG0F1R 71460800 IC50 = 1629 nM T99455 CZM79U 71460801 IC50 = 22.6 nM T99455 CWT1E8 71460802 IC50 = 0.69 nM T99455 CZ72YB 71460803 IC50 = 302 nM T99455 C8KL1P 71460845 IC50 = 1.42 nM T99455 C7XZ6K 71460846 IC50 = 66 nM T99455 CS08OH 71462551 IC50 = 0.45 nM T99455 CB45LP 71462552 IC50 = 0.41 nM T99455 C1IT5U 71550931 IC50 = 355 nM T99455 C5V8IC 71602940 IC50 = 4.73 nM T99455 C6SV9J 71602987 IC50 = 4125.31 nM T99455 CCQ25W 71602988 IC50 = 4.79 nM T99455 C6LKO2 71602989 IC50 = 3.21 nM T99455 C93MLS 71602992 IC50 = 34.77 nM T99455 CSP7K1 71603051 IC50 = 2754.9 nM T99455 CH7D8G 71603053 IC50 = 3.78 nM T99455 CHZ7U8 71603054 IC50 = 294.34 nM T99455 CWE69D 71603113 IC50 = 0.52 nM T99455 C4WT7O 71603114 IC50 = 2.34 nM T99455 CR08FQ 71603115 IC50 = 1.48 nM T99455 CE09DT 71603116 IC50 = 350.08 nM T99455 C4NM3G 71603117 IC50 = 1110.42 nM T99455 C62ZYM 71603170 IC50 = 63.31 nM T99455 CU8Z1W 71603171 IC50 = 6.34 nM T99455 CG80HO 73345816 IC50 = 199.53 nM T99455 CKA92Y 73348812 IC50 = 33189.45 nM T99455 CEUP75 73351906 IC50 = 50118.72 nM T99455 C7DSE2 73351907 IC50 = 10000 nM T99455 C8SUY0 73354884 IC50 = 398.11 nM T99455 CPJC10 73356444 IC50 = 1000 nM T99455 CCIS39 73356445 IC50 = 5370.32 nM T99455 C2PAK9 73438493 IC50 = 10 nM T99455 CHI51J 76070594 IC50 = 390 nM T99455 C8VAD5 76070929 IC50 > 10000 nM T99455 CB4V1R 76071142 IC50 = 380 nM T99455 CBAT06 76071144 IC50 = 89 nM T99455 C7SH1T 76071506 IC50 = 210 nM T99455 CS87EI 76071624 IC50 = 880 nM T99455 CGC0K4 76071869 IC50 > 10000 nM T99455 C9A8IG 79072608 IC50 = 255 nM T99455 CBP5K7 91183030 IC50 > 10000 nM T99455 CO07DQ 101879028 IC50 = 50 nM T99455 CG7YK9 101879029 IC50 = 17 nM T99455 CS8N1X 101879030 IC50 = 130 nM T99455 CUSN35 101879031 IC50 = 70 nM T99455 CY7BI2 118706214 IC50 > 10000 nM T99455 CDIA30 118722069 IC50 = 78600 nM T99455 C2SFD8 118722070 IC50 = 354000 nM T99455 C7CKE4 118722071 IC50 > 500000 nM T99455 C9ZW4S 118722072 IC50 = 385 nM T99455 CJPC58 118722073 IC50 > 500000 nM T99455 C53MDX 118722074 IC50 = 141000 nM T99455 CFC4T9 118722075 IC50 > 500000 nM T99455 CO9AY0 118722076 IC50 = 16100 nM T99455 C7YB8R 118722077 IC50 > 500000 nM T99455 CHD5Y4 118722078 IC50 = 6060 nM T99455 CIQ5K8 118722079 IC50 = 1440 nM T99455 C6CW9X 118722080 IC50 = 13500 nM T99455 C0M1KE 118722081 IC50 = 872 nM T99455 C5TD1S 118722083 IC50 = 277000 nM T99455 CF3YQ1 118722084 IC50 > 500000 nM T99455 CPR97Z 118722085 IC50 > 500000 nM T99455 CZ0I1M 118722086 IC50 = 91800 nM T99455 C2ACT5 118722089 IC50 > 500000 nM T99455 C5LBT6 118722090 IC50 = 563 nM T99455 CQ1S2N 118722091 IC50 = 266000 nM T99455 CQCX41 118737057 IC50 = 1 nM T99455 CUP4S1 122183740 IC50 = 14.2 nM T99455 CT12MC 122183741 IC50 = 15.9 nM T99455 CV3FM4 122183742 IC50 = 213.5 nM T99455 CVM71G 122183743 IC50 = 41.02 nM T99455 C48MKU 122183744 IC50 = 43.27 nM T99455 C2MK8C 122183745 IC50 = 46.2 nM T99455 CN3VR2 122183746 IC50 = 50.6 nM T99455 C43ELH 122183747 IC50 = 178 nM T99455 CG71PU 122183748 IC50 = 326 nM T99455 CUWG02 122183749 IC50 = 129.1 nM T99455 C6SQI8 122183750 IC50 = 26.58 nM T99455 C5X8JH 122183808 IC50 = 117.4 nM T99455 CG3ZX6 122183809 IC50 = 16.87 nM T99455 CM3NO8 122183810 IC50 = 175.3 nM T99455 C2P9NG 122186622 IC50 > 1000 nM T99455 CSVT14 122186623 IC50 = 300 nM T99455 C2V7EG 122189041 IC50 > 500000 nM T99455 C6MU0Y 122189043 IC50 = 66 nM T99455 C19CBJ 122189044 IC50 = 1156 nM T99455 CEQ5W9 122189045 IC50 = 45600 nM T99455 C5EX7F 122189047 IC50 = 276 nM T99455 C0JYX4 122189048 IC50 = 60670 nM T99455 C4UK5I 122189049 IC50 = 10220 nM T99455 CDT8R6 122189050 IC50 = 112 nM T99455 CR2Y7P 122189051 IC50 = 63300 nM T99455 C5OR0G 122189052 IC50 = 940 nM T99455 C82CRO 122189053 IC50 > 500000 nM T99455 CJ9HI8 122189054 IC50 = 19070 nM T99455 C9JI1S 122189056 IC50 > 500000 nM T99455 CYF0W2 122189057 IC50 = 143 nM T99455 C2YT3F 122189058 IC50 > 500000 nM T99455 CDY7N9 122189059 IC50 = 5050 nM T99455 C9Y5NU 122189060 IC50 = 89700 nM T99455 C54KBN 122189061 IC50 = 73 nM T99455 CR81XY 122189062 IC50 = 321 nM T99455 C4NK6A 122189064 IC50 = 444180 nM T99455 CO36WE 122189065 IC50 = 16 nM T99455 CL72TM 122189066 IC50 = 421 nM T99455 C6ZHF0 122189067 IC50 = 1837 nM T99455 CQ2SD8 122189068 IC50 > 500000 nM T99455 CDX9H3 122190820 IC50 = 2590 nM T99455 CSV74J 122190821 IC50 = 8530 nM T99455 C3ZQJ4 122190822 IC50 = 14550 nM T99455 C4AM5V 122190823 IC50 > 100000 nM T99455 CU3O4Q 122190824 IC50 = 9250 nM T99455 C4BL5S 122190825 IC50 = 11300 nM T99455 CZBP91 122190826 IC50 = 9240 nM T99455 C3PB0Z 122190828 IC50 = 4400 nM T99455 CT32LN 122190829 IC50 = 6200 nM T99455 C1EBW9 122190830 IC50 = 8960 nM T99455 CZ26FY 122190831 IC50 = 73910 nM T99455 C5Z2DL 122190832 IC50 = 35660 nM T99455 CW84RP 122190867 IC50 > 100000 nM T99455 CHU8E2 122190868 IC50 = 42170 nM T99455 CF2W4A 122190869 IC50 = 35040 nM T99455 CUP8H1 122190870 IC50 = 15320 nM T99455 CFR2Z0 122190871 IC50 = 51920 nM T99455 CV2N9D 122190872 IC50 > 100000 nM T99455 CL42TR 122190873 IC50 > 100000 nM T99455 C6QY7L 122196083 IC50 = 14 nM T99455 CP0WN2 122196084 IC50 = 86 nM T99455 CG48DP 122196085 IC50 = 49200 nM T99455 C0LWG4 122196086 IC50 = 3410 nM T99455 C0I6AZ 122196188 IC50 = 180 nM T99455 CJCH07 122196189 IC50 > 100000 nM T99455 CM0X4J 122196190 IC50 = 2760 nM T99455 CA8U7J 122196191 IC50 = 83520 nM T99455 C8LAJ2 122196192 IC50 > 100000 nM T99455 C47IXK 122196193 IC50 = 2370 nM T99455 C6BPW7 122196194 IC50 = 1890 nM T99455 CFE6L4 122196195 IC50 = 22760 nM T99455 CN4J5W 122196196 IC50 = 8560 nM T99455 CI9J5Z 122196197 IC50 = 75290 nM T99455 CU9V8Q 122196198 IC50 = 31 nM T99455 CL07SV 122196199 IC50 = 18 nM T99455 CWU4J7 122196200 IC50 = 56270 nM T99455 CRXT48 122196201 IC50 > 100000 nM T99455 CEQ32S 122196202 IC50 = 250 nM T99455 CS3U0R 122196203 IC50 > 100000 nM T99455 CQL0W7 122197565 IC50 > 10000 nM T99455 C6KM3T 127034964 EC50 = 1 nM T99455 C1BZ4L 127034965 EC50 = 3 nM T99455 C3IRJ0 127048197 IC50 > 10000 nM T99455 CZ07TW 127048198 IC50 > 10000 nM T99455 CS0H2C 127048199 IC50 > 10000 nM T99455 C1OE2F 127049532 IC50 = 580 nM T99455 C5P8TC 127049857 IC50 > 10000 nM T99455 CPQ35R 127049870 IC50 = 3880 nM T99455 CQO3X7 127049871 IC50 > 10000 nM T99455 C5H8LK 127051998 IC50 > 10000 nM T99455 CGT0B1 127052321 IC50 > 10000 nM T99455 C7NH6A 127052914 IC50 > 10000 nM T99455 CKB1Y6 127052915 IC50 > 10000 nM T99455 C6RPF1 130364436 IC50 > 10000 nM T99455 CSY34O 130364443 IC50 > 10000 nM T99455 CI9H2W 130364450 IC50 > 10000 nM T99455 CM4TO5 130364451 IC50 = 2100 nM T99455 CV4DH7 130364460 IC50 > 10000 nM T99455 CW91ZV 130364461 IC50 > 10000 nM T99455 CQIZ43 130364463 IC50 = 9900 nM T99455 C4IKC6 130364464 IC50 > 10000 nM T99455 C0X6JS 130364465 IC50 > 10000 nM T99455 C0ZGC1 130364467 IC50 > 10000 nM T99455 CO9C5Q 130364468 IC50 > 10000 nM T99455 CQW3P1 130364471 IC50 > 10000 nM T99455 CHWX05 130364473 IC50 = 8700 nM T99455 CLB65Y 130364478 IC50 = 4300 nM T99455 CUZG19 130364481 IC50 > 10000 nM T99455 C34OMJ 130364482 IC50 > 10000 nM T99455 C6TWR3 130364484 IC50 > 10000 nM T99455 C8SF5Q 130364488 IC50 = 547 nM T99455 CS5C4E 130364494 IC50 > 10000 nM T99455 CVQ32Y 130364503 IC50 > 10000 nM T99455 CV8B0Y 130364506 IC50 > 10000 nM T99455 CHX23J 130364524 IC50 = 10000 nM T99455 CHYL89 130364535 IC50 > 10000 nM T99455 CBI35E 132275094 IC50 = 942 nM T99455 CCG06O 134131688 IC50 = 122000 nM T99455 CFE03W 134131725 IC50 = 16200 nM T99455 CC3Y5M 134131924 IC50 = 320 nM T99455 C60IDE 134134575 IC50 = 220 nM T99455 C4TJD6 134135198 IC50 = 24 nM T99455 CUP01F 134135273 IC50 = 19 nM T99455 CKQV02 134135339 IC50 > 500000 nM T99455 CM3J8P 134137546 IC50 = 58000 nM T99455 C9QFX5 134139856 IC50 = 2280 nM T99455 C6Q9BT 134140130 IC50 = 15 nM T99455 CF0M3H 134140636 IC50 = 2580 nM T99455 C4AI2O 134141645 IC50 = 0.012 ug.mL-1 T99455 C0UT6Y 134141669 IC50 > 500000 nM T99455 CZA63L 134143363 IC50 = 1980 nM T99455 C3NS0E 134144264 IC50 = 19 nM T99455 CEU0N9 134144345 IC50 = 1440 nM T99455 C0R1TX 134144394 IC50 = 640 nM T99455 CF7KV6 134144611 IC50 = 1150 nM T99455 C18KJH 134145016 IC50 = 0.012 ug.mL-1 T99455 C35XCY 134145509 IC50 = 1690 nM T99455 C7W6PG 134147256 IC50 = 4520 nM T99455 C8AJ9S 134148237 IC50 = 2250 nM T99455 CJ7A2M 134148351 IC50 = 440 nM T99455 C8YCR0 134148385 IC50 = 19 nM T99455 CCL1G8 134148410 IC50 = 2650 nM T99455 C37NPG 134148847 IC50 = 385 nM T99455 CUL93K 134150012 IC50 > 500000 nM T99455 CI4EO5 134150056 IC50 > 500000 nM T99455 C1EY7B 134153245 IC50 = 890 nM T99455 CLC89D 134153463 IC50 = 0.012 ug.mL-1 T99455 CFTL08 134155527 IC50 = 560 nM T99455 CAOK49 134155843 IC50 > 500000 nM T99455 CX6Q8G 134157397 IC50 > 500000 nM T99455 CQR94G 134198433 IC50 > 10000 nM T99455 C46QAS 135441185 EC50 = 10 nM T99455 C0PVG7 135819982 EC50 = 360 nM T99455 C2PJK6 135820173 EC50 = 70 nM T99455 C53LFX 135820297 EC50 = 970 nM T99455 CP7KZ8 135820466 EC50 = 1800 nM T99455 CQK62L 135820498 EC50 = 560 nM T99455 C4PD2G 135820511 EC50 = 30 nM T99455 CDT7E4 136211077 IC50 > 100 nM T99455 C5VE4K 137636547 IC50 > 10000 nM T99455 CZ05TY 137637593 IC50 > 10000 nM T99455 C6PKY7 137645383 IC50 > 10000 nM T99455 CHR9E0 137651685 IC50 = 414 nM T99455 CY53VO 137651787 IC50 > 10000 nM T99455 CE8DW7 137658399 IC50 > 10000 nM T99455 CU61WM 137658936 IC50 > 10000 nM T99455 CY9N8Q 137662234 IC50 = 8100 nM T99455 C0PYR1 138454771 EC50 < 10 nM T99455 CO9P7G 145351804 IC50 > 1000 nM T99455 CBR08X 145983359 IC50 = 1107 nM T99455 CE2X6V 145983518 IC50 = 435 nM T99455 C4ID8J 145984666 IC50 = 211 nM T99455 CD49VM 155295006 IC50 > 10000 nM T99455 CA8IF5 155510457 IC50 = 10660 nM T99455 CSHC63 155510467 IC50 > 10000 nM T99455 CG09WO 155512858 IC50 > 10000 nM T99455 C6H8ZU 155513172 IC50 = 2220 nM T99455 COI8N1 155513641 IC50 = 3720 nM T99455 CZDH58 155514096 IC50 > 10000 nM T99455 CEB08Z 155514919 IC50 = 6280 nM T99455 C84GJO 155517474 IC50 > 10000 nM T99455 CHQ5X7 155518340 IC50 = 6230 nM T99455 CP1B5K 155518600 IC50 = 520 nM T99455 C63PZX 155518871 IC50 > 10000 nM T99455 CC1A2U 155518947 IC50 = 4280 nM T99455 C1U3HE 155522045 IC50 = 110 nM T99455 C8EZ6J 155523550 IC50 = 31610 nM T99455 CF72IY 155527080 IC50 = 17560 nM T99455 CITV17 155527171 IC50 = 5750 nM T99455 C8DF2W 155529116 IC50 = 2160 nM T99455 CNP8T7 155530083 IC50 = 237 nM T99455 CK10UA 155531677 IC50 = 3696 nM T99455 C54ARD 155532371 IC50 = 170 nM T99455 C4DT6V 155532665 IC50 = 2340 nM T99455 CWLZ25 155535008 IC50 > 10000 nM T99455 C8NA6L 155536370 IC50 = 437 nM T99455 CL9X4S 155540971 IC50 = 2450 nM T99455 C3Q9UA 155541932 IC50 > 10000 nM T99455 CI27QV 155546853 IC50 > 10000 nM T99455 CYP2O5 155547984 IC50 = 1452 nM T99455 CB85AE 155550823 IC50 = 380 nM T99455 CL8KR2 155552517 IC50 = 989.3 nM T99455 C1TA9J 155553503 IC50 > 10000 nM T99455 CJS68O 155553593 IC50 = 290 nM T99455 C8BAU3 155554243 IC50 > 10000 nM T99455 CCQF25 155555943 IC50 > 10000 nM T99455 C9QM2K 155559937 IC50 = 1500 nM T99455 CN9LE6 155560662 IC50 = 5850 nM T99455 CHLY93 155562871 IC50 = 5345 nM T99455 C60KLJ 155564326 IC50 = 4992 nM T99455 C4BS6J 155565938 IC50 = 5637 nM T99455 CINX89 155566065 IC50 = 5120 nM T99455 CVMG35 155566307 IC50 = 1350 nM T99455 C7Q4RY 155566792 IC50 = 1813 nM T99455 CP69SU 155567937 IC50 > 10000 nM T99455 C8VT6Z 155568644 IC50 = 1990 nM T99455 D00AII 5281727 IC50 = 10000 nM T99455 D03EHM 24905142 IC50 = 18 nM T99455 D03NPX 447077 IC50 = 2 nM T99455 D03PLP 11579996 IC50 = 8000 nM T99455 D05UJT 5311510 EC50 = 140 nM T99455 D05XGZ 11536458 IC50 = 42000 nM T99455 D08RZB 11153014 IC50 = 3 nM T99455 D0AW4W 11537051 IC50 = 6000 nM T99455 D0AZ0Y 11514345 IC50 = 20000 nM T99455 D0H4YH 11594901 IC50 = 10000 nM T99455 D0I3XZ 11601743 IC50 = 4200 nM T99455 D0N7AJ 11409972 IC50 = 580 nM T99455 D0O9NE 5388063 IC50 = 10000 nM T99455 D0PI0R 11609210 IC50 = 14000 nM T99455 D0QG6G 11493254 IC50 = 14000 nM T84631 D05EAM 4735 IC50 = 10400 nM T84631 D05PHH 3447 IC50 = 4610 nM T84631 D07UWV 92722 Ki = 53000 nM T84631 D07XHO 4413 IC50 = 21100 nM T84631 D0I0RJ 16231 IC50 > 50000 nM T84631 D0I5HF 10182969 Ki = 0.08 nM T84631 D0J0BU 10275777 Ki = 0.117 nM T84631 D0KG3R 9875401 Ki = 0.4 nM T84631 D0M7JT 216210 Ki > 1000 nM T84631 D00LOB 9866964 Ki = 3300 nM T84631 D01MUU 183797 Ki = 3680 nM T84631 D05TKW 16098914 IC50 = 1900 nM T84631 D07BRZ 9939865 Ki = 4.6 nM T84631 D07KWN 99514 Ki = 13385 nM T84631 D0I7MX 9871765 Ki = 22.5 nM T84631 D0ID3W 9911502 Ki = 4 nM T84631 D0PK7J 56599309 Ki = 206 nM T84631 D0X2NN 9826322 IC50 = 2.7 nM T84631 D02INZ 2387 IC50 = 4500 nM T84631 D02MHE 9806376 IC50 = 301 nM T84631 D02QTV 122267 IC50 = 16 nM T84631 D03QJN 9895762 Ki = 0.15 nM T84631 D0D5RH 11641515 Ki = 1.8 nM T84631 D0E2MJ 5496659 Ki = 0.4 nM T84631 D0J9UI 9807238 Ki = 1.3 nM T84631 D0K1PR 1747 Ki = 22000 nM T84631 D0N7WR 108040 Ki = 20400 nM T84631 D0S2JG 9913629 Ki = 1100 nM T84631 D0T4UL 11634458 IC50 = 0.57 nM T84631 CR8YG3 1308 Ki = 34 nM T84631 C71WRJ 1503 Ki = 8900 nM T84631 CY5B9C 1504 Ki = 2100 nM T84631 C2KE5Q 1508 Ki = 2700 nM T84631 C4S1PB 4300 Ki = 115000 nM T84631 CL1T7V 4301 Ki = 12000 nM T84631 C8D4SG 5107 Ki = 0.9 nM T84631 C2OG9Z 47978 IC50 = 100 nM T84631 CMG15V 122129 Ki = 7 nM T84631 CS5RN9 178051 Ki = 47973.34 nM T84631 CZP0Y1 204101 Ki = 0.19 nM T84631 CM32OH 402499 IC50 > 50000 nM T84631 C4Q9XJ 402501 IC50 > 50000 nM T84631 C3YP0R 444562 Ki = 26000 nM T84631 C3R5AJ 445480 Ki = 22 nM T84631 CRN1F6 445481 Ki = 18 nM T84631 C2Z0XW 445482 Ki = 0.7 nM T84631 CR4KE5 445844 Ki = 19000 nM T84631 CU6X2A 445847 Ki = 31000 nM T84631 CI64QU 446399 IC50 = 33 nM T84631 CHD15V 446604 Ki = 38018.94 nM T84631 C9GU2P 446605 Ki = 42657.95 nM T84631 C7IE4P 446606 Ki = 20989.4 nM T84631 C4M8WT 446979 Ki = 28 nM T84631 CS4OB0 446982 Ki = 25 nM T84631 C5E3YX 446984 Ki = 9 nM T84631 C17BWY 447193 Ki = 0.76 nM T84631 CM3T9E 447194 Ki = 0.059 nM T84631 CZC4U1 447359 Ki = 4 nM T84631 CNO6G5 447360 Ki = 1.1 nM T84631 C85OTU 447361 Ki = 3 nM T84631 C9QXV5 447362 Ki = 1 nM T84631 C5UX1L 447478 Ki = 990 nM T84631 CVND42 447482 Ki = 2400 nM T84631 C4OKV5 447486 Ki = 34000 nM T84631 CC9G5O 447490 Ki = 34000 nM T84631 CR2DX3 447496 Ki = 300 nM T84631 COYS31 447502 Ki = 6800 nM T84631 CVI28M 447508 Ki = 52 nM T84631 CS09BE 447510 Ki = 570 nM T84631 C87GLP 447540 Ki = 65000 nM T84631 C6FD5N 447889 Ki = 15135.61 nM T84631 CK9Q4X 448061 Ki = 13 nM T84631 C43LRO 448062 Ki = 1.6 nM T84631 COK45L 448065 Ki = 0.27 nM T84631 CFMI91 448548 Ki = 3000 nM T84631 CSL82K 449091 Ki = 26000 nM T84631 COK61H 639391 Ki = 0.66 nM T84631 C9D4IN 754821 IC50 > 50000 nM T84631 CB5C6X 1034712 IC50 = 4224 nM T84631 C1CNZ9 2756474 Ki = 680000 nM T84631 CER5L6 2796875 Ki = 11 nM T84631 CO4K7H 3037565 IC50 = 11418 nM T84631 C24VNC 3083488 Ki = 41020.41 nM T84631 C0K7TF 3123858 IC50 > 50000 nM T84631 C8KD9E 3162843 IC50 > 50000 nM T84631 CQ6N8P 3496895 Ki = 13 nM T84631 CT8JE1 4655928 Ki = 1400 nM T84631 CZEI30 5282448 IC50 = 11 nM T84631 C0KI2N 5287439 Ki = 0.1 nM T84631 CPZ6A3 5287506 Ki = 8000 nM T84631 C48TEQ 5287836 Ki = 13 nM T84631 CQ26VM 5289531 Ki = 15000 nM T84631 C1B9GP 5400404 IC50 > 50000 nM T84631 C0CV5L 5496928 IC50 = 270 nM T84631 CAW1P7 5497056 Ki = 0.9 nM T84631 C7SYK9 6102731 IC50 = 35 nM T84631 C5YL6I 6420136 Ki = 18 nM T84631 C2ZRF5 6540265 Ki = 3 nM T84631 C5XV7G 6540266 Ki = 0.07 nM T84631 CY1J7X 6540267 Ki = 89 nM T84631 CN57IY 6540268 Ki = 3 nM T84631 C8MS7Y 6852168 Ki = 6 nM T84631 CN2B6S 6852211 Ki = 10000 nM T84631 C49IOZ 6857707 Ki = 140000 nM T84631 CM8R6E 6914706 IC50 = 160 nM T84631 CNZA87 9112697 IC50 > 200000 nM T84631 CX34ZD 9549214 Ki = 0.14 nM T84631 CME7Y3 9549257 Ki = 90 nM T84631 CXY5Z7 9549258 Ki = 15 nM T84631 CYRC97 9549259 Ki = 47 nM T84631 CAE25N 9549260 Ki = 1 nM T84631 CK64FD 9794516 IC50 >= 10300 nM T84631 CJ52KF 9794796 IC50 = 90000 nM T84631 CVFE34 9800775 IC50 = 1190 nM T84631 C92QSE 9801235 IC50 > 100000 nM T84631 C2FHU7 9801905 IC50 = 640 nM T84631 C3CL2G 9803364 Ki = 11 nM T84631 C4VX9Y 9803558 Ki = 8 nM T84631 CTA52P 9803848 Ki > 15000 nM T84631 C8QGS1 9804434 Ki = 16 nM T84631 CDN8P2 9804727 Ki = 103000 nM T84631 C1FIN6 9804775 IC50 > 130 nM T84631 C4OTK6 9805415 Ki = 1.9 nM T84631 CAKN38 9805632 Ki = 3.8 nM T84631 C6JIT7 9806444 IC50 = 3300 nM T84631 CBKL18 9806644 IC50 = 13 nM T84631 CW3NK6 9806974 Ki = 9.5 nM T84631 CKP97L 9807142 Ki = 1.2 nM T84631 CX1C7P 9807257 Ki = 260 nM T84631 C6F3XK 9807686 Ki = 43 nM T84631 CS62VX 9808020 IC50 = 0.83 nM T84631 CAG59M 9808035 Ki = 47 nM T84631 CTS98Y 9808170 Ki = 4.9 nM T84631 CH9IE6 9808346 IC50 = 2.3 nM T84631 CZS3H5 9808724 Ki = 3400 nM T84631 C2AXV0 9809479 Ki = 1.1 nM T84631 C60AVD 9812184 Ki = 910 nM T84631 CLTO67 9821317 IC50 > 100000 nM T84631 C4KEZ2 9821506 Ki > 500 nM T84631 CNCV95 9823140 IC50 = 1708 nM T84631 CJ2G7A 9823668 IC50 = 21 nM T84631 CX6DA7 9823789 Ki = 1600 nM T84631 CD3AP6 9824122 Ki = 198 nM T84631 CZ64PW 9824925 Ki = 164 nM T84631 C1YZP2 9825165 Ki = 39 nM T84631 CTG89N 9825830 Ki = 5 nM T84631 CPB20R 9826345 Ki = 3 nM T84631 CKH36Z 9826433 IC50 = 12 nM T84631 CS1DL7 9826716 IC50 = 3.6 nM T84631 CYR35V 9827147 IC50 = 34 nM T84631 CB82VS 9827306 Ki = 5.7 nM T84631 CK5VW1 9827389 IC50 = 3.9 nM T84631 CA7W3I 9827682 IC50 = 13 nM T84631 C6J0KE 9827723 Ki = 600 nM T84631 CGN48U 9827867 IC50 = 6000 nM T84631 CEJ3D7 9827921 Ki = 38 nM T84631 CVP0C6 9828249 IC50 = 15 nM T84631 CGD13M 9828337 IC50 = 14 nM T84631 CB65VJ 9828393 Ki = 10 nM T84631 CE0HD3 9828470 Ki = 84800 nM T84631 CRH01E 9828697 Ki = 500 nM T84631 C9A5SY 9828818 Ki = 21978.6 nM T84631 COW7Q3 9829120 Ki = 1.3 nM T84631 CP2X5B 9829453 Ki = 28 nM T84631 C7BW5P 9829585 Ki < 0.1 nM T84631 C5RVZ4 9829804 Ki = 62 nM T84631 C8RV5E 9830070 Ki = 500 nM T84631 C4F8CN 9830285 IC50 = 1410 nM T84631 C4T5BQ 9830932 Ki = 360 nM T84631 CH38SL 9840270 Ki = 220 nM T84631 CVO5R3 9842851 IC50 = 1370 nM T84631 C53JFK 9844392 Ki = 19 nM T84631 CC4Y8V 9845104 Ki = 275 nM T84631 C6VAG8 9845526 IC50 = 84 nM T84631 C2TA1I 9845742 IC50 > 30000 nM T84631 CM8Y9G 9846259 IC50 = 10000 nM T84631 C8I4LS 9846496 Ki = 900 nM T84631 CM0OU9 9847373 IC50 > 2500 nM T84631 CU2H1W 9848037 IC50 = 120 nM T84631 C5Z2RH 9848091 IC50 = 104 nM T84631 CSQ8V7 9848265 IC50 = 7.3 nM T84631 CX25MR 9848465 Ki = 0.5 nM T84631 CW3EC6 9848592 Ki = 5300 nM T84631 CCL5G3 9848846 IC50 = 0.55 nM T84631 C80PNB 9849423 IC50 = 1.6 nM T84631 CS9HQ0 9850467 IC50 = 19.3 nM T84631 CH9L1I 9850515 Ki = 1.8 nM T84631 CEQ92L 9850889 IC50 = 1.6 nM T84631 CR7S2O 9851195 Ki = 1.1 nM T84631 CP8CY7 9859977 IC50 > 200000 nM T84631 CRTD24 9863579 Ki = 55000 nM T84631 CB86RC 9864323 Ki = 50 nM T84631 CF74PR 9864759 IC50 = 1120 nM T84631 C89JRZ 9868633 Ki = 8300 nM T84631 CQ5J9K 9868873 Ki = 0.1 nM T84631 CL6QS0 9868922 Ki = 2100 nM T84631 CDVE40 9869375 Ki = 0.78 nM T84631 C5A1LI 9870767 IC50 = 4.5 nM T84631 C38BTY 9870834 Ki = 0.75 nM T84631 CZ9LR2 9870910 Ki = 4500 nM T84631 C1AW6N 9870947 Ki = 20 nM T84631 CIL85V 9871029 IC50 = 38 nM T84631 C9UB6X 9871197 Ki = 3.5 nM T84631 CX51SZ 9871369 IC50 = 1.6 nM T84631 CHP0C8 9872347 Ki = 400 nM T84631 CIZ61P 9872423 Ki > 75400 nM T84631 C6ZB3K 9872552 IC50 = 18 nM T84631 CG0L6A 9873029 IC50 = 3.2 nM T84631 CAJ92Z 9873782 Ki = 22 nM T84631 C5LV1Z 9873979 IC50 = 6000 nM T84631 CPU3D1 9881263 IC50 > 200000 nM T84631 CS78YB 9882885 IC50 > 200000 nM T84631 C2F5NS 9884570 Ki = 1300 nM T84631 C83BSN 9885116 Ki = 4200 nM T84631 CQP0V2 9886960 Ki = 460 nM T84631 CJT9X7 9887558 Ki = 102 nM T84631 C6A4TL 9890540 Ki = 11 nM T84631 C17NPU 9890541 IC50 = 20.9 nM T84631 CC3R5Y 9890878 Ki = 0.18 nM T84631 CO4QD2 9891154 Ki = 3.4 nM T84631 C7E1IV 9891337 IC50 = 20.6 nM T84631 CT6W0R 9891759 Ki = 4400 nM T84631 CD13TH 9891795 IC50 > 10000 nM T84631 C80RWQ 9892098 Ki = 1.9 nM T84631 C1M2PU 9892103 IC50 = 3510 nM T84631 C8UV6Y 9892106 Ki = 0.33 nM T84631 C79RJF 9892295 IC50 = 750 nM T84631 C7I5RG 9892392 Ki = 16000 nM T84631 CG5VS0 9892818 IC50 = 29 nM T84631 C6QE7Y 9893007 IC50 > 11000 nM T84631 CKN8D4 9893040 Ki = 92 nM T84631 CXY68Z 9893122 IC50 = 337 nM T84631 CNJ0W1 9893177 IC50 = 1390 nM T84631 C4A6TQ 9893238 Ki = 3 nM T84631 C5IG2W 9893544 Ki = 0.32 nM T84631 C4DHN5 9894203 Ki = 1.5 nM T84631 CB4O8L 9894223 Ki = 2.7 nM T84631 C13KVD 9894553 Ki = 2000 nM T84631 CCSP64 9894606 Ki = 170 nM T84631 CKDP84 9895193 Ki = 1700 nM T84631 CZY9L0 9905436 IC50 = 174000 nM T84631 C0SP6Q 9906596 Ki = 120 nM T84631 C2HN7L 9907201 Ki = 42 nM T84631 C85SEZ 9908687 IC50 > 10000 nM T84631 CMC95R 9910164 Ki = 165 nM T84631 CAP0O8 9910540 Ki = 50 nM T84631 CD5LQ0 9910982 Ki > 15000 nM T84631 CAWD59 9911275 IC50 = 30 nM T84631 CS6QF5 9912191 Ki > 30000 nM T84631 C75QYP 9912650 IC50 = 5.8 nM T84631 CJ5Y8N 9912741 IC50 = 20 nM T84631 C0LKE7 9912771 Ki = 31 nM T84631 C8GJF3 9913055 IC50 = 39.6 nM T84631 CU94XJ 9913274 IC50 = 95 nM T84631 C4N0IJ 9913371 IC50 = 10 nM T84631 CUF7C2 9913912 IC50 = 9.9 nM T84631 C49HMD 9914510 Ki = 1.7 nM T84631 C1C3VT 9914538 IC50 = 11 nM T84631 CUVX26 9914911 Ki = 360 nM T84631 CC0D5H 9915041 Ki = 0.91 nM T84631 CPZ50Y 9915193 Ki = 0.29 nM T84631 CVND52 9915545 Ki > 10000 nM T84631 C2GWH3 9916339 Ki = 71 nM T84631 CX45DI 9916346 Ki = 1760 nM T84631 CH8QJ4 9916876 Ki = 0.014 nM T84631 CHG59Y 9916885 Ki = 330 nM T84631 C0Z3HS 9917367 IC50 = 39 nM T84631 CK2H1C 9917705 Ki = 0.52 nM T84631 CF9SD1 9917846 IC50 = 2 nM T84631 CFO1K9 9922130 Ki > 1000000 nM T84631 CLZ53G 9922131 Ki > 1000000 nM T84631 CAP64B 9929157 Ki = 9 nM T84631 C2TO4N 9931543 Ki = 2900 nM T84631 C9I2ES 9931785 IC50 = 1500 nM T84631 CY0TP3 9932394 IC50 = 20 nM T84631 CI8JS1 9933581 IC50 = 24 nM T84631 C7H6NL 9933675 IC50 = 8 nM T84631 C85LIU 9934003 Ki = 0.15 nM T84631 CS9Y5I 9934133 IC50 = 7200 nM T84631 C7V9BM 9934351 Ki = 4 nM T84631 CLT7P8 9934591 IC50 = 2 nM T84631 CSY16U 9934960 Ki = 11.5 nM T84631 C38QWF 9935364 Ki = 0.06 nM T84631 CG3B1P 9935390 Ki = 0.5 nM T84631 C1XT2Y 9935746 Ki = 2 nM T84631 CL2NV0 9935925 IC50 > 870 nM T84631 C5KS0R 9936020 IC50 = 6 nM T84631 CKLJ26 9936190 IC50 > 100000 nM T84631 C49DRC 9936691 IC50 = 376 nM T84631 CL0U1E 9936850 IC50 = 0.5 nM T84631 CDT2W8 9936861 Ki = 2.8 nM T84631 CG96QC 9936983 Ki = 3.9 nM T84631 COA4R0 9937032 Ki = 2.3 nM T84631 C07XOI 9937041 Ki = 29 nM T84631 CC9QH7 9937406 IC50 = 270 nM T84631 CK76DL 9937410 Ki = 10 nM T84631 C8F5CW 9937921 Ki = 0.15 nM T84631 C8LR4T 9938917 Ki = 1.7 nM T84631 CNE34O 9939021 IC50 = 1 nM T84631 CDT95S 9939426 Ki = 980 nM T84631 C1RHT8 9949886 Ki = 210 nM T84631 CD27EJ 9951054 IC50 = 66 nM T84631 CP06LN 9953722 Ki = 15 nM T84631 CD7ZO5 9954791 Ki = 3.9 nM T84631 C0R4GE 9954812 IC50 = 7.5 nM T84631 CX85LD 9954980 Ki = 0.43 nM T84631 CK9N1A 9955155 IC50 = 0.9 nM T84631 CP7A2W 9955292 Ki = 1200 nM T84631 CSI62L 9955475 IC50 = 851 nM T84631 C3EPC4 9955758 Ki > 22000 nM T84631 CV96ZD 9955999 Ki = 110 nM T84631 C58QTM 9956404 Ki = 1 nM T84631 CY5OI8 9956416 IC50 = 5000 nM T84631 C8Y4EG 9956632 Ki = 16 nM T84631 CW4SU3 9956768 Ki = 7500 nM T84631 CI84CP 9957386 Ki = 0.35 nM T84631 CN36AS 9957822 Ki = 0.63 nM T84631 C85CTV 9957994 IC50 = 646 nM T84631 CLM2E6 9958023 Ki = 150 nM T84631 CE39JM 9958168 Ki = 3900 nM T84631 CU2YV0 9958249 IC50 = 7.8 nM T84631 C76ZFQ 9958477 Ki = 1300 nM T84631 CRM6L7 9958614 IC50 = 11 nM T84631 CLW0D4 9959111 IC50 = 3 nM T84631 C2Y0QV 9959268 IC50 = 3.4 nM T84631 CEHA54 9959604 IC50 = 2.1 nM T84631 CX59ZG 9959715 Ki = 350 nM T84631 CBC2K3 9959749 IC50 = 0.8 nM T84631 C0C1FQ 9959919 Ki = 1.5 nM T84631 COMH01 9961613 Ki = 1.7 nM T84631 C0TV8Q 9962561 Ki >= 200000 nM T84631 CTMU52 9978512 IC50 = 200 nM T84631 C3BNE7 9979006 IC50 = 1015 nM T84631 C3S7IV 9979724 Ki = 262 nM T84631 CV81FG 9980363 IC50 = 500 nM T84631 C38MBH 9981197 Ki = 0.07 nM T84631 C4CH0E 9981449 Ki = 99000 nM T84631 CWGL23 9982191 Ki = 130 nM T84631 C6XM2Z 9982428 Ki = 0.041 nM T84631 CK6XE9 9982431 IC50 > 30000 nM T84631 CY3Z7I 9982644 IC50 = 170 nM T84631 C5SA7F 9983043 IC50 > 2500 nM T84631 C5UGC0 9983309 Ki = 0.046 nM T84631 CCP75S 9983704 Ki = 6.4 nM T84631 C59OAZ 9983994 IC50 = 5.3 nM T84631 CZ50EY 9984282 IC50 = 1.9 nM T84631 C0OA9T 9984718 Ki = 270 nM T84631 CIP45F 9984838 IC50 = 3.5 nM T84631 CZ6TD1 9985759 Ki = 21 nM T84631 CKP2Z7 9987204 Ki > 33700 nM T84631 CKIP10 9987251 IC50 = 79000 nM T84631 CEC95B 9997816 Ki = 400 nM T84631 CE75GM 10000477 IC50 = 640 nM T84631 CJ0Q2S 10002821 Ki = 6 nM T84631 CVQN23 10003356 Ki = 11 nM T84631 C56FZK 10003877 IC50 = 15000 nM T84631 C4KCS7 10004019 Ki = 3600 nM T84631 CU9QI6 10004529 Ki = 0.037 nM T84631 C9O5SJ 10004800 Ki = 0.77 nM T84631 CH5BV6 10005347 Ki = 29991.63 nM T84631 C8I7YZ 10006319 IC50 = 200 nM T84631 CZJ38W 10006399 IC50 > 25000 nM T84631 CR34FA 10007463 Ki = 0.14 nM T84631 CFQV59 10007890 Ki = 2.4 nM T84631 CGL95Q 10008517 Ki = 3890.45 nM T84631 C7Q8PK 10009640 Ki = 0.016 nM T84631 CB1SY8 10023491 IC50 = 1700 nM T84631 C8ME3O 10024183 Ki = 7 nM T84631 CBM0Q3 10026319 Ki = 0.048 nM T84631 CF1V4K 10027758 Ki = 3 nM T84631 CW5JH1 10028252 Ki = 0.9 nM T84631 C3SU6O 10028986 Ki = 0.4 nM T84631 CX4TI5 10029172 Ki = 340 nM T84631 C3E4DR 10029213 IC50 = 6700 nM T84631 C4PFW9 10029239 Ki = 0.55 nM T84631 CI2O5B 10029343 Ki = 1.1 nM T84631 CB4Y7M 10030046 IC50 = 24 nM T84631 CTO52N 10030167 Ki = 5 nM T84631 CDL3M7 10030847 Ki = 8 nM T84631 C5LQ4A 10032429 Ki = 1.7 nM T84631 CUG6R3 10037159 Ki = 27 nM T84631 CSX68Z 10043156 IC50 = 1100 nM T84631 CK4W6M 10047815 IC50 = 52000 nM T84631 C3DIK1 10048418 IC50 = 61 nM T84631 C9R8YW 10048823 Ki = 50.5 nM T84631 C8FKM2 10049151 IC50 = 39000 nM T84631 CILJ89 10050878 IC50 = 28 nM T84631 C80QYS 10051154 Ki = 92000 nM T84631 C08PUS 10051441 IC50 = 81 nM T84631 CVY28G 10051489 Ki = 4.2 nM T84631 C29DTM 10051582 Ki = 0.2 nM T84631 CU9I7D 10051599 Ki = 12 nM T84631 CHZL08 10051960 Ki = 3.4 nM T84631 C3QP6V 10052373 Ki = 54 nM T84631 CXL9H7 10052619 Ki = 51 nM T84631 COP2U4 10052951 Ki = 3 nM T84631 CFCT67 10053115 Ki = 0.5 nM T84631 CDE42G 10053298 Ki = 5500 nM T84631 CXZ2V3 10054210 Ki = 1.3 nM T84631 C1OI8R 10066101 Ki = 4600 nM T84631 C6F4SZ 10067786 Ki = 12 nM T84631 CBV7N2 10070407 IC50 = 4100 nM T84631 CW28HS 10071127 Ki = 11 nM T84631 CI2KG6 10072299 IC50 > 30000 nM T84631 CP65QI 10073006 Ki = 0.023 nM T84631 CV5F8U 10073425 Ki = 3.3 nM T84631 C7TU4O 10073666 Ki = 0.6 nM T84631 CB04YW 10073864 IC50 > 100000 nM T84631 CF4R2W 10074230 IC50 = 260 nM T84631 CF18ZA 10074434 Ki = 2.8 nM T84631 CUOC38 10074752 Ki = 4.7 nM T84631 CAT42M 10074892 Ki > 300000 nM T84631 C9ZCS2 10074922 IC50 = 1600 nM T84631 CF0R6D 10074927 IC50 > 25000 nM T84631 C2CUX3 10075442 Ki = 1.8 nM T84631 COL31T 10075735 Ki = 0.1 nM T84631 C46JXH 10076965 IC50 = 72 nM T84631 CD0VO9 10078364 IC50 = 27 nM T84631 CR0ZL7 10091675 IC50 = 1600 nM T84631 CP38MH 10091962 IC50 = 1500 nM T84631 CPY49G 10092707 IC50 = 11750 nM T84631 CZM79H 10093390 Ki > 15000 nM T84631 C4P3ZO 10093667 IC50 = 15000 nM T84631 C3TDM1 10094168 Ki = 5 nM T84631 C2VT9U 10094219 Ki = 0.5 nM T84631 CZH3W7 10094378 Ki = 160000 nM T84631 C0FS4U 10094458 IC50 = 840 nM T84631 CMHD92 10094532 IC50 = 66000 nM T84631 CRXD40 10095024 Ki = 2800 nM T84631 CQP65H 10095093 Ki = 3600 nM T84631 C6PVA7 10095315 IC50 = 530 nM T84631 C3TWI1 10095455 Ki = 1 nM T84631 C3OG5U 10095865 Ki = 2 nM T84631 C0JE3C 10096795 IC50 = 150 nM T84631 C3XBN4 10097126 IC50 = 27 nM T84631 C8L7HY 10097631 Ki = 2330 nM T84631 C3IRT4 10098156 Ki = 5400 nM T84631 CRS8D1 10098302 Ki = 2.2 nM T84631 C6V2QM 10098361 Ki = 0.11 nM T84631 COSB36 10098572 Ki = 0.02 nM T84631 C9TN8U 10098702 Ki = 380 nM T84631 CD3VB0 10099008 Ki = 0.074 nM T84631 CX8A6G 10099038 Ki > 8000 nM T84631 CO8G7N 10099218 IC50 = 2 nM T84631 CP39AO 10099570 IC50 = 4.8 nM T84631 CO7J9C 10099638 Ki = 26 nM T84631 CV6NQ3 10099674 Ki > 8000 nM T84631 CW6IS3 10113744 IC50 = 20 nM T84631 C7HKG1 10114497 IC50 < 0.5 nM T84631 CH4Z6B 10116752 Ki = 0.14 nM T84631 CW4RZ5 10116936 IC50 > 450 nM T84631 C1VT4F 10117027 Ki = 15 nM T84631 C9V2WC 10117161 IC50 = 52 nM T84631 CK69GS 10117541 Ki = 0.24 nM T84631 CXCR46 10117543 Ki > 75000 nM T84631 C1XZ8N 10117556 IC50 = 4 nM T84631 CM34QP 10118017 Ki = 4 nM T84631 CL9RB8 10118144 Ki = 0.28 nM T84631 CB4QC8 10118358 Ki = 0.97 nM T84631 C9PG6D 10119254 Ki = 0.001 nM T84631 CX9VL6 10119957 Ki = 300 nM T84631 CV5E4L 10121049 Ki > 75400 nM T84631 C4TB7E 10121121 Ki = 15 nM T84631 CL68QZ 10121795 IC50 = 128 nM T84631 CS32UJ 10128374 Ki = 0.3 nM T84631 C3JPD6 10128550 Ki = 44.5 nM T84631 C1BA9E 10128598 Ki = 2 nM T84631 CJP02S 10128788 Ki = 5.3 nM T84631 C6AET3 10128907 Ki = 19 nM T84631 C0KQ9U 10129004 Ki = 2 nM T84631 C4FV1T 10129354 Ki = 1 nM T84631 CR03NV 10131788 Ki > 1000000 nM T84631 CN9F5G 10137016 Ki = 0.044 nM T84631 CJYD93 10137523 IC50 = 187 nM T84631 C7QB2E 10138114 IC50 = 32 nM T84631 CUCF82 10139899 Ki = 0.97 nM T84631 CVA35H 10140425 Ki = 178.6 nM T84631 CMFW67 10140911 Ki = 0.51 nM T84631 C67VZS 10141105 IC50 = 2 nM T84631 CF68DH 10141182 Ki = 3 nM T84631 CWF4I3 10141502 Ki = 5400 nM T84631 CN2WO7 10141594 Ki = 2.8 nM T84631 C1Q3KU 10141691 Ki = 0.73 nM T84631 CRH46O 10142203 Ki = 0.013 nM T84631 C1SKF3 10142819 IC50 = 6.7 nM T84631 C17YOT 10142920 Ki = 2 nM T84631 C54YQM 10143087 IC50 = 1320 nM T84631 C31QAL 10143532 Ki = 0.21 nM T84631 CYCG10 10151574 Ki = 24 nM T84631 CJ52ND 10152434 Ki = 2 nM T84631 C6XYM8 10152710 Ki = 11 nM T84631 CJ93LZ 10152785 Ki = 7 nM T84631 C86MJA 10152813 Ki = 1 nM T84631 C7HW4S 10161422 IC50 = 90 nM T84631 C95PMZ 10161902 IC50 = 26 nM T84631 CVZ23C 10162019 Ki = 53 nM T84631 C5IQ3M 10162145 IC50 = 1.5 nM T84631 C4K3WG 10162441 Ki = 96.4 nM T84631 CV27BE 10162765 Ki = 189 nM T84631 CT65YJ 10162799 Ki = 5300 nM T84631 CBHY78 10163266 Ki = 248.6 nM T84631 CF82TK 10163421 Ki = 6.3 nM T84631 C75ADN 10164065 Ki = 0.92 nM T84631 CM6PS4 10165173 Ki = 111000 nM T84631 C1QBH5 10165288 Ki = 11 nM T84631 C5WB4J 10165649 Ki > 75400 nM T84631 C7G4JC 10166616 Ki > 75400 nM T84631 CEPJ05 10166622 Ki > 75400 nM T84631 C5I0YH 10168444 Ki = 20 nM T84631 C24FCQ 10174464 Ki = 2 nM T84631 CD60LF 10174479 Ki = 6.8 nM T84631 CG2B8A 10174487 Ki = 15 nM T84631 CHPZ12 10174488 Ki = 3 nM T84631 CL0BI3 10174813 Ki = 78 nM T84631 CB17JX 10174938 Ki = 19 nM T84631 CMX71K 10174991 Ki = 2 nM T84631 C86UTO 10175171 Ki = 3 nM T84631 COVN41 10175189 Ki = 6.9 nM T84631 CG37YX 10181104 IC50 > 30000 nM T84631 CN2ZL1 10182437 IC50 = 8.2 nM T84631 COD9C2 10183134 IC50 = 3 nM T84631 CX9NV0 10183250 Ki = 16 nM T84631 CF4S8B 10183471 Ki = 0.6 nM T84631 CT31ZH 10183608 Ki = 152.7 nM T84631 CM0X5B 10184785 Ki = 1.4 nM T84631 C5K2GS 10185181 IC50 = 1.3 nM T84631 C7PC2K 10185292 IC50 > 170 nM T84631 CK5WD2 10185323 Ki = 15 nM T84631 C93EKT 10185327 Ki = 76.8 nM T84631 C3U1NL 10185372 Ki = 600 nM T84631 CTA49K 10185508 IC50 = 12 nM T84631 CFIH78 10185526 IC50 = 100 nM T84631 C7U3IT 10185995 Ki = 0.057 nM T84631 CU24HL 10186048 Ki = 16 nM T84631 C14TNW 10187006 Ki = 1 nM T84631 C1DN4F 10187311 Ki = 82100 nM T84631 CZ9KS7 10188952 Ki = 46 nM T84631 CG9T8S 10189755 IC50 = 1548 nM T84631 CKI5B8 10195400 Ki = 11 nM T84631 CK2Z4I 10195824 Ki = 7 nM T84631 C4P6BM 10195843 Ki = 2 nM T84631 CE3PG5 10196628 Ki = 81 nM T84631 CY5XQ6 10196732 Ki = 1 nM T84631 CO6VM1 10196955 Ki = 7396.05 nM T84631 CF2E6U 10198683 IC50 = 32000 nM T84631 CZ09JV 10202260 IC50 = 4 nM T84631 CHY62J 10203373 Ki = 2.9 nM T84631 CCV6X8 10203976 IC50 = 0.8 nM T84631 CO51ZR 10205659 Ki = 0.06 nM T84631 C2CWI1 10206231 Ki = 370 nM T84631 CFS69U 10206365 Ki = 2.4 nM T84631 CO4QT2 10207346 IC50 = 3250 nM T84631 COY39X 10207569 IC50 = 6.7 nM T84631 CW62PU 10207853 Ki = 1.6 nM T84631 CRL6T9 10207889 IC50 = 8.7 nM T84631 CT0S2D 10208075 Ki = 5 nM T84631 C1H2FS 10208201 Ki = 0.3 nM T84631 C01QTR 10209142 Ki > 75400 nM T84631 CP69QR 10212999 IC50 = 80 nM T84631 C7FTD2 10217291 Ki = 200 nM T84631 C1YOJ4 10217652 Ki = 5 nM T84631 CJRS38 10217801 Ki = 3 nM T84631 C42CUP 10217822 Ki = 370 nM T84631 CML04S 10218126 Ki = 6 nM T84631 C0DPK8 10218244 Ki = 4.8 nM T84631 CG8NY9 10218368 Ki = 73 nM T84631 C3P2VS 10218446 Ki = 2 nM T84631 CG7OS8 10225234 IC50 = 1.4 nM T84631 C6HAC0 10227428 Ki = 0.98 nM T84631 CM8O7V 10227632 Ki = 10 nM T84631 CYR45Q 10227730 IC50 > 30000 nM T84631 CIAX57 10228506 Ki > 75000 nM T84631 CSR74M 10228660 IC50 > 100000 nM T84631 CN1PX4 10228720 Ki = 29 nM T84631 CY41MS 10228870 Ki = 10 nM T84631 C98FSX 10230007 Ki = 103000 nM T84631 CMU21W 10231661 Ki = 85200 nM T84631 C87QYI 10239204 Ki = 350 nM T84631 C7G5XE 10239342 Ki = 0.17 nM T84631 CX3DY4 10239377 Ki = 2 nM T84631 CEM6N7 10239497 Ki = 1 nM T84631 C2O5HU 10239546 Ki = 53 nM T84631 CD0X3A 10239600 Ki = 23988.33 nM T84631 CSM4Y6 10239728 Ki = 4 nM T84631 CF4ND2 10247830 Ki = 5600 nM T84631 C9QML3 10250104 Ki = 57 nM T84631 CCI28E 10250490 Ki = 1.5 nM T84631 CC04IK 10253196 IC50 = 1010 nM T84631 C7RVY1 10253674 Ki = 15 nM T84631 CG8MU6 10254797 Ki = 1.5 nM T84631 C4Z1LU 10255253 Ki = 12 nM T84631 C71RTC 10255760 IC50 = 5.2 nM T84631 CS4F5P 10256448 IC50 > 100000 nM T84631 CD6V5R 10256934 IC50 = 27 nM T84631 C4WV1A 10257345 IC50 = 0.83 nM T84631 CFBN38 10257580 IC50 = 30 nM T84631 CJN34G 10258080 Ki = 0.037 nM T84631 C91KHA 10258902 Ki = 0.02 nM T84631 CVJ0I9 10258984 Ki = 0.013 nM T84631 CAM06S 10273747 IC50 = 43 nM T84631 CYZ79T 10274887 IC50 = 140 nM T84631 CQ9ZO1 10275412 Ki = 0.11 nM T84631 C50WLH 10278497 IC50 = 4 nM T84631 CL7E8K 10280735 Ki = 0.56 nM T84631 CB1S5P 10281431 Ki > 75400 nM T84631 CSEV08 10289091 Ki = 0.25 nM T84631 CMP9A5 10289373 Ki = 260 nM T84631 CXL1S0 10289409 Ki = 75000 nM T84631 C5BRU4 10289601 Ki = 13 nM T84631 CCV2P1 10289690 Ki = 28 nM T84631 CS8E7Y 10289697 Ki = 1999.86 nM T84631 CK2R3I 10290214 Ki = 0.88 nM T84631 CZM97W 10293977 Ki = 110000 nM T84631 C0T3CN 10296435 IC50 > 100000 nM T84631 CT2A4B 10297501 IC50 = 8 nM T84631 CV10CU 10297977 Ki = 0.044 nM T84631 CM62FC 10298615 IC50 = 4060 nM T84631 C1AP6H 10298858 Ki = 0.105 nM T84631 C79BFH 10298942 Ki = 0.09 nM T84631 C03FHY 10299568 IC50 = 2 nM T84631 CPX8N9 10299701 Ki = 0.23 nM T84631 CDP9R7 10299889 Ki = 29 nM T84631 CLJ02I 10300491 Ki = 0.47 nM T84631 CDY8F9 10300557 Ki = 1100 nM T84631 CEW97F 10301102 Ki = 3000 nM T84631 C6JSB5 10301730 Ki = 3 nM T84631 C29IBW 10303308 IC50 = 6.2 nM T84631 CGTF74 10303947 Ki > 75400 nM T84631 C17RDU 10304095 Ki > 10000 nM T84631 C8PA9J 10310498 Ki = 8 nM T84631 C0PQ6I 10311006 Ki = 4 nM T84631 CVYT89 10311026 Ki = 6 nM T84631 C4DQJ1 10311346 Ki = 2600 nM T84631 CU4HS2 10311517 Ki = 11 nM T84631 CHGS42 10311669 Ki = 9 nM T84631 C9N1TU 10311760 Ki < 1 nM T84631 CFTS84 10311761 Ki = 5 nM T84631 CN8FL2 10315612 Ki = 970 nM T84631 CMR75W 10318568 IC50 > 100000 nM T84631 C25XSY 10318999 IC50 = 4100 nM T84631 CGO0R3 10321806 IC50 = 60 nM T84631 C8Y4EJ 10322243 Ki > 15000 nM T84631 CMR6Y8 10323469 Ki = 1.6 nM T84631 CC7LN6 10324201 Ki = 0.05 nM T84631 C8SQ1N 10324263 IC50 = 8 nM T84631 CX9J5U 10324635 Ki = 3.7 nM T84631 C6QPK0 10324772 Ki = 100 nM T84631 CT0FX4 10325259 Ki > 8000 nM T84631 C56PEV 10325271 IC50 > 2500 nM T84631 CJ28HS 10325481 Ki = 1.8 nM T84631 CA67OL 10325720 Ki = 730 nM T84631 C41ZLB 10326602 IC50 = 4.9 nM T84631 C53QGN 10339033 Ki > 15000 nM T84631 CN5R3I 10340020 Ki = 400 nM T84631 CZMH83 10340538 IC50 = 45000 nM T84631 C4YR1M 10342318 Ki = 12000 nM T84631 CP64HV 10342843 Ki = 980000 nM T84631 C30ODG 10342944 IC50 = 1948 nM T84631 CV8J6G 10343097 Ki = 7 nM T84631 CKSH17 10343499 IC50 = 85 nM T84631 CFL57Y 10343633 Ki = 0.44 nM T84631 CK9J7X 10343728 Ki = 154 nM T84631 C4I7DQ 10345176 Ki = 0.026 nM T84631 C8FO7Q 10345230 Ki = 0.035 nM T84631 CES6C2 10345244 Ki = 5900 nM T84631 CT9GJ0 10345579 Ki = 1.1 nM T84631 CGBX39 10346320 Ki < 0.02 nM T84631 CH0RW2 10346646 IC50 = 490 nM T84631 CZ2WV3 10347131 Ki = 23 nM T84631 C3ZS2H 10347405 Ki = 1 nM T84631 C4KER5 10347610 IC50 = 18.7 nM T84631 CI4LG1 10347624 Ki = 1.8 nM T84631 CL09QG 10349678 IC50 = 290 nM T84631 C83DLG 10361934 Ki = 0.66 nM T84631 CL07UC 10364218 Ki > 10000 nM T84631 C1XV4P 10364890 IC50 = 2794 nM T84631 CW29YO 10365461 IC50 = 310 nM T84631 CH0V8B 10366070 Ki = 13 nM T84631 C0ODK9 10366157 IC50 = 16000 nM T84631 C0XW1E 10366176 IC50 = 360 nM T84631 CO0Z6Y 10366592 Ki = 1.8 nM T84631 C10ISY 10367012 Ki = 95000 nM T84631 CJ0O5P 10367277 IC50 > 33000 nM T84631 CIQ63E 10367299 IC50 = 230 nM T84631 CG98CM 10367552 Ki = 0.7 nM T84631 C5T6DO 10367956 Ki = 0.75 nM T84631 CJWE07 10368488 IC50 = 190 nM T84631 CDO83F 10368538 Ki > 75000 nM T84631 C5PR3L 10368553 Ki = 2.5 nM T84631 C9ZD0S 10368685 Ki = 0.46 nM T84631 CNV3A1 10369141 Ki = 0.055 nM T84631 CE27CV 10370457 Ki = 4400 nM T84631 C6HML8 10371129 Ki = 0.043 nM T84631 CYBF76 10386378 Ki = 6.9 nM T84631 C26CSM 10386393 IC50 = 2200 nM T84631 C71PIO 10387118 Ki > 20 nM T84631 C7TH5Q 10387956 Ki = 3 nM T84631 CMNP39 10389039 Ki = 0.7 nM T84631 CLGF71 10389462 Ki = 9 nM T84631 CE45NM 10389524 Ki = 0.16 nM T84631 CL3F1U 10389579 Ki = 2.5 nM T84631 CM6L0W 10389769 Ki > 10000 nM T84631 C4ITG3 10389930 Ki = 1 nM T84631 C47OZV 10390121 Ki = 1.2 nM T84631 C3BR5A 10390490 Ki = 2.4 nM T84631 CXF20B 10391310 IC50 = 3000 nM T84631 CJNV62 10391699 IC50 > 33000 nM T84631 C6S4CO 10391715 Ki = 8 nM T84631 CEH4D1 10391881 Ki = 14 nM T84631 CLK08Z 10391999 Ki = 0.8 nM T84631 CNS5B3 10392083 Ki = 5 nM T84631 CF6P1M 10392348 Ki = 3500 nM T84631 C94IOU 10392838 Ki = 2 nM T84631 C6QP4U 10393267 Ki = 0.1 nM T84631 CCA45U 10394183 IC50 = 59 nM T84631 CM1WJ6 10394292 Ki = 12 nM T84631 C4FBO0 10409093 Ki = 12 nM T84631 C56NXW 10409551 IC50 = 12000 nM T84631 CO3Z5D 10409945 IC50 = 1700 nM T84631 CMQY61 10410471 Ki > 15000 nM T84631 C2L8SQ 10410499 IC50 = 4200 nM T84631 C9AM3R 10410743 IC50 = 11000 nM T84631 CL34IB 10410866 Ki = 60000 nM T84631 C70AME 10411443 IC50 = 130000 nM T84631 C7K8JS 10411444 IC50 = 2218 nM T84631 C20ZSL 10411684 Ki = 0.32 nM T84631 CD0VI1 10412365 Ki = 18 nM T84631 C03MWI 10413130 Ki = 10 nM T84631 CF8M6C 10415115 Ki = 3050 nM T84631 CVK4L6 10418061 IC50 > 100000 nM T84631 CS4DL8 10433086 Ki = 13 nM T84631 C1RE8V 10433463 IC50 = 0.18 nM T84631 C4K9QX 10433872 IC50 = 9500 nM T84631 CFIC58 10434349 Ki = 0.041 nM T84631 CK3YW7 10434792 Ki = 0.087 nM T84631 C6L5IM 10434906 Ki = 1.6 nM T84631 C6AZ8B 10435038 Ki = 500 nM T84631 CX39AB 10435238 Ki = 18 nM T84631 CHCI84 10435532 Ki > 15000 nM T84631 CUM2T7 10436294 Ki = 2.5 nM T84631 C46YOA 10437408 IC50 = 5.8 nM T84631 C4L9EK 10438017 Ki = 650 nM T84631 CG07WY 10438196 Ki = 0.15 nM T84631 CL4K2S 10447733 IC50 = 112000 nM T84631 CCU35L 10453208 IC50 = 700000 nM T84631 C9M5RI 10453763 Ki > 15000 nM T84631 C4SZV0 10454685 Ki > 10000 nM T84631 C7HOX3 10454867 IC50 = 1000 nM T84631 CV9N1X 10457101 Ki = 7.2 nM T84631 C4M7SR 10458428 IC50 = 19 nM T84631 C50FMX 10458597 Ki = 550 nM T84631 C7M5HE 10459832 Ki = 0.079 nM T84631 C9W5IS 10460210 Ki = 5800 nM T84631 C9HI6A 10460541 IC50 = 1.9 nM T84631 CI87FD 10460564 IC50 = 1.2 nM T84631 CKM0N3 10460673 IC50 = 4 nM T84631 C7O6BE 10477973 Ki = 47 nM T84631 C53XJD 10478176 Ki = 560 nM T84631 C0W7NM 10478661 Ki > 15000 nM T84631 C63GRO 10479438 IC50 = 328 nM T84631 C1MX6F 10480245 Ki > 15000 nM T84631 C45KWI 10480373 Ki = 0.7 nM T84631 CCP2N8 10480374 Ki = 21 nM T84631 CV0X6G 10480463 IC50 = 0.2 nM T84631 CN1YX8 10480534 Ki = 0.074 nM T84631 CF2G8Q 10481025 Ki = 9 nM T84631 CM5A3J 10481558 Ki = 0.1 nM T84631 CMIN26 10481978 Ki = 0.32 nM T84631 CKIQ80 10482395 Ki = 0.054 nM T84631 CJ50AY 10483408 Ki = 10 nM T84631 CEI65Z 10483775 Ki = 340 nM T84631 CKL8H3 10497634 Ki = 230 nM T84631 CQE12B 10501172 Ki = 52 nM T84631 C1F7IZ 10501283 Ki = 24400 nM T84631 C6F2ZX 10501400 Ki = 52 nM T84631 CFU1E5 10501943 Ki = 110 nM T84631 CFP53Y 10502109 IC50 > 33000 nM T84631 CKI70V 10502393 Ki = 98 nM T84631 CEKX36 10503075 Ki = 1300 nM T84631 C4O9JK 10503954 Ki = 140 nM T84631 CY16UR 10504366 Ki = 1100 nM T84631 C0U6NB 10504802 Ki = 38500 nM T84631 CG5IS0 10505288 Ki = 0.005 nM T84631 C09TUO 10506433 Ki = 21 nM T84631 CXB50R 10508061 Ki = 66 nM T84631 CQS6Y2 10523322 Ki = 200 nM T84631 CFL49H 10524222 Ki = 1800 nM T84631 C87BCM 10525391 Ki = 700 nM T84631 CJ15UC 10525392 Ki = 11900 nM T84631 CD82SZ 10525943 Ki = 130 nM T84631 CZ0E8S 10526100 Ki = 34 nM T84631 C42XPE 10526785 Ki = 240 nM T84631 C7Y0WM 10527751 Ki = 41 nM T84631 CS7UC4 10528210 Ki = 280 nM T84631 CU8I0J 10528552 Ki = 4.1 nM T84631 CT41XW 10528653 Ki = 190 nM T84631 CF1PZ4 10530789 IC50 = 2000 nM T84631 CA0QG6 10531178 Ki = 0.8 nM T84631 C1K0NS 10532026 Ki = 53 nM T84631 CKYZ01 10532259 Ki = 4.2 nM T84631 C7S9QW 10532670 IC50 = 30 nM T84631 COB07E 10543987 Ki > 30000 nM T84631 CK13IY 10546004 Ki = 550 nM T84631 CO1JW8 10546322 Ki = 420 nM T84631 CEP1L6 10547293 Ki = 140 nM T84631 CO46GQ 10548215 Ki = 29000 nM T84631 CYEN07 10548429 Ki = 600 nM T84631 CEC7J6 10549325 Ki = 2200 nM T84631 C2F6CT 10549508 Ki = 12 nM T84631 CB81VQ 10551446 Ki = 440 nM T84631 CDH1F3 10552170 Ki = 440 nM T84631 CVR3P1 10552445 Ki = 130 nM T84631 C4Q5VT 10552446 IC50 = 0.008 nM T84631 CYX1V7 10553919 Ki = 9.4 nM T84631 C4J1KI 10554052 Ki = 919 nM T84631 CE8V0B 10555065 Ki = 220 nM T84631 CWR8G9 10555769 Ki = 130 nM T84631 CGQ38W 10555959 Ki = 380 nM T84631 CQG10I 10556031 Ki = 21 nM T84631 CSK8V5 10556085 Ki = 6.8 nM T84631 CGHL47 10556206 Ki = 4.3 nM T84631 CY1JF2 10569959 Ki = 940 nM T84631 CZ6HD9 10570938 Ki = 1642 nM T84631 C52FQT 10571832 Ki = 192 nM T84631 C1HA7S 10572228 Ki = 12 nM T84631 C2VG9M 10572774 Ki = 1.3 nM T84631 CV71RX 10573919 Ki = 620 nM T84631 CS8H3A 10574097 Ki = 59 nM T84631 CSHM62 10575806 Ki = 78 nM T84631 CY5O2K 10576002 Ki = 110 nM T84631 CY1A0X 10576138 Ki = 330 nM T84631 C9MN1H 10579028 Ki = 890 nM T84631 C6LO8Q 10580222 Ki = 0.32 nM T84631 C1D8GI 10580396 Ki = 0.44 nM T84631 C42LVU 10580437 Ki = 3.5 nM T84631 C02RYN 10592155 Ki = 5000 nM T84631 C4VMO3 10595198 Ki = 2800 nM T84631 CWJ68A 10596601 Ki = 95 nM T84631 CO3N1I 10597592 Ki > 10000 nM T84631 CI5CH1 10597827 Ki = 0.46 nM T84631 CT2E6F 10598802 Ki = 2.5 nM T84631 CJZF07 10599669 Ki = 7000 nM T84631 C7SEQ9 10599734 Ki = 2600 nM T84631 CD6L3E 10600145 Ki = 1100 nM T84631 CCQU28 10600245 Ki = 3.1 nM T84631 C8L9FV 10600329 Ki = 1200 nM T84631 CVEH84 10600484 Ki = 240000 nM T84631 C0SD6T 10603555 Ki = 1600 nM T84631 CP69LR 10604270 Ki = 68 nM T84631 C8CQY2 10604382 Ki < 5 nM T84631 CY1J0N 10604774 Ki = 2.1 nM T84631 C1RH3P 10621200 Ki = 654 nM T84631 CC26YF 10622456 Ki > 5000 nM T84631 CO83BP 10622800 IC50 = 120 nM T84631 C39IFP 10623057 Ki = 180 nM T84631 C5K8QJ 10623402 Ki > 100000 nM T84631 CXD95O 10623670 Ki = 720 nM T84631 CSP20T 10623756 Ki = 83 nM T84631 CZJL67 10623842 Ki = 7 nM T84631 CV0I5Y 10623890 Ki = 41 nM T84631 C3OJ4U 10623965 Ki = 0.04 nM T84631 C69VAT 10624206 Ki = 6 nM T84631 C1ZW5F 10624489 Ki = 100 nM T84631 C8SUZ9 10624948 Ki = 640 nM T84631 C8S6QZ 10625945 Ki = 1300 nM T84631 C8PHU2 10626697 Ki = 27000 nM T84631 CJ62ZG 10626722 Ki > 100000 nM T84631 CK25AY 10626893 Ki = 160000 nM T84631 CQ7F0T 10627268 Ki = 480 nM T84631 C03CIN 10628066 Ki = 2.4 nM T84631 C1PX0H 10642149 Ki = 18 nM T84631 CF3P4J 10642387 Ki = 53 nM T84631 C4KMJ8 10644692 Ki = 390 nM T84631 CZ9L8T 10644693 Ki = 18 nM T84631 C4M0QB 10645022 Ki = 140 nM T84631 C0QP4O 10645136 Ki = 9900 nM T84631 C3S0GW 10645345 Ki = 640 nM T84631 CFNH06 10645807 IC50 = 53 nM T84631 C72XTB 10646342 Ki = 225 nM T84631 CNC25X 10646757 Ki = 130 nM T84631 CRMG36 10647285 Ki = 1000 nM T84631 C1XDA6 10647609 IC50 = 950 nM T84631 CR1Y2D 10647704 Ki = 2.3 nM T84631 C76RFN 10647907 Ki = 22 nM T84631 CR5EX8 10648196 Ki = 820 nM T84631 C41KHW 10648454 Ki = 4 nM T84631 C1KVB3 10650805 Ki > 200000 nM T84631 C2OSA9 10651120 Ki > 100000 nM T84631 C6E4WZ 10651873 Ki = 2.2 nM T84631 CG40SW 10661464 Ki = 5100 nM T84631 CRDG85 10665326 Ki = 130 nM T84631 C4WCH6 10668443 Ki = 660 nM T84631 CUD8A7 10669525 Ki = 1100 nM T84631 C7CVW2 10669933 IC50 = 240 nM T84631 CD2C0U 10670479 Ki = 5.2 nM T84631 C6PAD8 10670666 Ki = 500 nM T84631 CZO1K8 10671210 Ki = 210 nM T84631 C4LJO3 10671702 Ki > 100000 nM T84631 CIKJ09 10672223 Ki = 7 nM T84631 CW1G9B 10672666 IC50 > 10000 nM T84631 CP6RF7 10673965 IC50 = 333 nM T84631 CM1Y2D 10675086 Ki = 62 nM T84631 C4TIU1 10675632 Ki = 0.008 nM T84631 C8P2UC 10675884 Ki = 8.8 nM T84631 CFQ5V2 10690751 Ki = 1850 nM T84631 CVE95Z 10691360 Ki = 24 nM T84631 CI48CW 10692578 Ki = 230 nM T84631 CD8S2B 10692579 Ki = 60 nM T84631 C4KBY2 10692711 IC50 = 6216 nM T84631 CID1F6 10693808 Ki > 33700 nM T84631 CZ53XC 10693841 Ki > 5000 nM T84631 CS08UM 10694720 Ki = 690 nM T84631 CVR1F9 10694772 Ki = 160 nM T84631 CIB63V 10694800 Ki = 3.1 nM T84631 C5VB1U 10695159 Ki = 8700 nM T84631 C2W4YZ 10695208 Ki = 220 nM T84631 CW8RV0 10696389 Ki = 8 nM T84631 CP4QC5 10696511 Ki > 1000000 nM T84631 C3QH0L 10697320 Ki = 5 nM T84631 C3WC0Q 10698376 Ki = 230000 nM T84631 CWX87E 10698758 Ki > 100000 nM T84631 C4B1DG 10712659 Ki > 5000 nM T84631 CY0P5F 10714145 Ki = 220 nM T84631 CF6TZ2 10715258 Ki = 1150 nM T84631 CK2WI6 10715476 Ki = 59 nM T84631 CZB24K 10715861 Ki = 280 nM T84631 C0TE1Z 10716448 Ki = 2400 nM T84631 C49JDV 10717698 Ki = 3300 nM T84631 CFG6T3 10717789 Ki = 100 nM T84631 CPGV87 10718240 Ki = 18000 nM T84631 CCP58N 10718840 Ki = 3.4 nM T84631 C82FPL 10718889 Ki = 120 nM T84631 CFH75T 10718950 Ki = 380 nM T84631 C1Z3PF 10719336 Ki = 0.007 nM T84631 COA5Z1 10719523 Ki = 43 nM T84631 CIKF89 10719580 Ki = 220000 nM T84631 CLXN90 10721219 Ki = 41 nM T84631 CM58XP 10721501 IC50 = 700 nM T84631 CMUX37 10722043 Ki = 240 nM T84631 CAS17I 10722747 Ki = 0.8 nM T84631 CUTA38 10723163 Ki = 0.92 nM T84631 CF9VZ0 10738109 Ki > 500 nM T84631 CZ0G6W 10738922 Ki = 130 nM T84631 C1GCY4 10739768 Ki = 2.8 nM T84631 CL7RC5 10742017 IC50 > 33000 nM T84631 C64AUD 10742143 Ki = 150 nM T84631 CK26FW 10742542 Ki = 11 nM T84631 C5L7HE 10745242 Ki > 100000 nM T84631 CAUM51 10745299 Ki = 0.01 nM T84631 CU5OG9 10746409 Ki = 6780 nM T84631 C8C1BP 10746437 Ki = 74131.02 nM T84631 C3V8JP 10746573 Ki = 0.06 nM T84631 C8J9PM 10761427 Ki = 22900 nM T84631 C9JLQ7 10761484 Ki = 2400 nM T84631 CHA46Q 10764382 Ki > 500 nM T84631 C0FTS9 10764466 Ki = 32 nM T84631 C9SDJ1 10765420 Ki = 120 nM T84631 CD51XL 10765919 Ki = 130 nM T84631 CQUM96 10765972 Ki = 370 nM T84631 C2YPX5 10766061 Ki = 0.047 nM T84631 CJSW62 10767268 Ki = 150 nM T84631 CKOQ35 10767421 Ki = 7100 nM T84631 C9SQB5 10767957 Ki = 0.009 nM T84631 CCK3E5 10768801 Ki = 8 nM T84631 C5DYQ3 10769476 Ki = 2.7 nM T84631 C62KFB 10769759 Ki = 4.1 nM T84631 C24ZSE 10769921 Ki = 11 nM T84631 C5E6AY 10770527 Ki = 2.9 nM T84631 C4Z2LQ 10770606 Ki = 1.7 nM T84631 CQW74C 10770621 Ki = 1.6 nM T84631 CCZ9U0 10770773 Ki = 1 nM T84631 C3W7TF 10770845 Ki = 1.7 nM T84631 C7VXA1 10784195 Ki = 2800 nM T84631 CJ7O1H 10785523 Ki = 5.6 nM T84631 CI9BZ1 10786604 Ki = 42 nM T84631 CQRZ02 10787180 Ki = 320 nM T84631 CD1CF3 10787181 Ki = 350 nM T84631 C0AUV8 10788046 Ki > 5000 nM T84631 C4CAT2 10788047 Ki = 4.8 nM T84631 CRHE34 10788206 Ki = 190 nM T84631 CD21MW 10788364 Ki = 9800 nM T84631 CKLU46 10788963 Ki = 395 nM T84631 C0RL4C 10789777 Ki = 250 nM T84631 CMX5V9 10789805 Ki = 970 nM T84631 CT8M1C 10790019 Ki = 310 nM T84631 CL73OX 10791003 Ki = 160000 nM T84631 C5TID3 10791816 Ki = 120 nM T84631 CBNP58 10792157 Ki = 56 nM T84631 CRD65S 10792619 Ki > 200000 nM T84631 CLWY92 10793236 Ki = 14000 nM T84631 C5ENU2 10794450 Ki = 0.11 nM T84631 C64ZVF 10794532 Ki = 4.2 nM T84631 CC95IV 10794535 Ki = 8.5 nM T84631 CD6U1P 10806942 Ki = 1400 nM T84631 CR51LN 10807566 Ki = 4579 nM T84631 CYAJ14 10810195 Ki = 4.6 nM T84631 CL9O0C 10810196 Ki = 500 nM T84631 CUQX02 10810754 Ki = 340 nM T84631 C74QCG 10811600 Ki = 1200 nM T84631 C0U7PJ 10811747 Ki = 510 nM T84631 CYS08X 10813043 Ki = 14 nM T84631 CQK97I 10813230 Ki = 49 nM T84631 C3WX4F 10813359 Ki = 2.4 nM T84631 C13KAX 10813709 Ki = 70 nM T84631 CZA0D1 10814968 Ki = 0.02 nM T84631 CE1DT2 10815540 Ki = 25 nM T84631 CV1U5L 10816337 Ki = 31 nM T84631 CL8YB0 10816451 Ki = 34 nM T84631 CPRS52 10817210 Ki = 7600 nM T84631 CSZR21 10817699 Ki = 9.9 nM T84631 CUS6D0 10818009 Ki = 19 nM T84631 C0M3XB 10831506 Ki = 53 nM T84631 C9HPZ8 10831834 IC50 = 6300 nM T84631 CE2LP4 10832026 Ki > 5000 nM T84631 CLXP56 10833102 Ki = 1400 nM T84631 C6NW5I 10833234 Ki > 5000 nM T84631 CJ2M4I 10835535 Ki = 23 nM T84631 CW8OT1 10835646 Ki = 110 nM T84631 C2KXJ7 10835995 Ki = 750 nM T84631 CH0RG9 10836919 Ki = 570 nM T84631 C67FIC 10837478 Ki = 55 nM T84631 CW3YA2 10837929 Ki = 120 nM T84631 C1FTR2 10837980 Ki = 6 nM T84631 C5FSB0 10838473 Ki = 62 nM T84631 CM13CR 10840852 Ki = 0.6 nM T84631 CYX51H 10840933 Ki = 7.2 nM T84631 CZVR32 10841125 Ki = 10000 nM T84631 COLC79 10841532 Ki = 52000 nM T84631 C6QF7T 10841535 Ki = 17800 nM T84631 C2R7OQ 10841758 Ki = 3.3 nM T84631 CJRU60 10860637 Ki = 948 nM T84631 CBK06L 10861643 IC50 > 60000 nM T84631 C6F2ZP 10863119 Ki = 10000 nM T84631 C7U4IT 10863260 Ki = 1720 nM T84631 CB38YZ 10863406 Ki > 5000 nM T84631 CK7VC8 10863579 Ki = 820 nM T84631 C07BLI 10864217 Ki = 50 nM T84631 C62IPV 10864710 Ki = 11 nM T84631 C02XLH 10865109 IC50 = 240 nM T84631 CZX59B 10865289 Ki = 14 nM T84631 C9LEJ0 10865386 IC50 = 1700 nM T84631 C1BOZ5 10865461 IC50 = 270 nM T84631 CN2CE8 10865462 IC50 = 610 nM T84631 CLB15C 10871563 Ki > 75000 nM T84631 CWVZ13 10873723 Ki = 262 nM T84631 CD7I4A 10873871 Ki = 1800 nM T84631 CPSW72 10873946 Ki = 45 nM T84631 C0KIZ5 10874086 Ki = 220 nM T84631 CXG62W 10874449 Ki = 38 nM T84631 C3Z6PT 10874628 IC50 > 30000 nM T84631 C2TH3I 10875009 Ki = 154 nM T84631 C7YEP4 10875960 IC50 = 2400 nM T84631 C80WCU 10883641 Ki = 1700 nM T84631 CTAF76 10884388 Ki = 19 nM T84631 CAR7T6 10884739 Ki = 5310 nM T84631 CZP9L7 10884798 Ki = 1556 nM T84631 CJWL05 10884908 Ki = 798 nM T84631 C1PNQ4 10885181 Ki > 5000 nM T84631 C27LWG 10885612 Ki = 99 nM T84631 C8EG3O 10886723 Ki = 226 nM T84631 CK6T4L 10892244 Ki = 10000 nM T84631 CCA1Q7 10894246 Ki = 6890 nM T84631 CU8J0C 10894269 Ki = 28 nM T84631 CNL3H2 10894415 Ki = 2000 nM T84631 CJGS43 10894874 Ki = 26 nM T84631 CW9MC1 10894892 Ki = 5800 nM T84631 C49BRD 10894895 Ki = 320 nM T84631 CW7Q2U 10895700 IC50 > 250000 nM T84631 C16NXJ 10896126 Ki = 13 nM T84631 CKY20H 10896140 Ki > 5000 nM T84631 CMP45U 10896308 Ki = 2700 nM T84631 C1YPJ0 10896662 Ki = 42 nM T84631 C39AVR 10897080 Ki = 7 nM T84631 C59ETF 10897550 Ki = 23 nM T84631 C2GPU4 10897682 IC50 = 1030 nM T84631 CQTC02 10903566 Ki = 6800 nM T84631 C8J1TX 10904089 Ki <= 11000 nM T84631 CR9G0E 10905722 Ki = 1200 nM T84631 CB1HW4 10905809 IC50 > 30000 nM T84631 C1F8UV 10905825 Ki = 3600 nM T84631 C9C6UE 10906426 Ki = 600 nM T84631 CH2G5Q 10906977 Ki > 75000 nM T84631 CTM36K 10907121 Ki = 5500 nM T84631 C3FY5S 10907552 Ki = 133 nM T84631 CPJ1Q7 10908669 IC50 = 160 nM T84631 C9E7RY 10908791 IC50 = 1250 nM T84631 C2BXU9 10908808 IC50 = 300 nM T84631 C5I7SU 10916321 Ki = 530 nM T84631 CA1IB4 10916653 Ki = 4000 nM T84631 CX3FP2 10917491 Ki > 5000 nM T84631 C7K5SQ 10918066 Ki = 160 nM T84631 COQY14 10918387 Ki = 2064 nM T84631 CCDO06 10919424 Ki = 84 nM T84631 C5A8NU 10919581 IC50 = 570 nM T84631 CMK60F 10927859 Ki = 720 nM T84631 CKI49C 10928313 Ki = 21000 nM T84631 CR5VW1 10928435 Ki = 15 nM T84631 CMK6P8 10928757 IC50 > 30000 nM T84631 CK6E0Q 10928936 Ki = 840 nM T84631 C7Z6JY 10929059 Ki = 6790 nM T84631 C1KV7H 10929853 Ki = 28 nM T84631 CT5H0B 10929908 Ki = 50 nM T84631 C1Q9WZ 10930326 IC50 = 2120 nM T84631 CL20KX 10930722 IC50 = 1070 nM T84631 CG7NA5 10938859 Ki > 1200 nM T84631 C8RF5U 10938960 Ki = 500 nM T84631 CMD6C0 10939317 Ki = 26 nM T84631 CC81OU 10939381 Ki = 1300 nM T84631 CT4G3S 10939409 Ki = 2700 nM T84631 CDSU98 10939678 Ki > 5000 nM T84631 C3MY5I 10940389 Ki = 85 nM T84631 CG5BN9 10940660 Ki = 160 nM T84631 CSZX24 10941224 Ki = 24 nM T84631 C5ED3R 10946700 Ki = 7910 nM T84631 C8OA1L 10946869 Ki = 43000 nM T84631 CUN98K 10949030 Ki = 1350 nM T84631 C3NR1O 10949672 Ki = 131 nM T84631 CCM7H1 10949960 Ki = 400 nM T84631 CJDM01 10950292 Ki = 2400 nM T84631 C95WOX 10950363 Ki = 1800 nM T84631 CUWF38 10950398 Ki = 68 nM T84631 CWN81P 10950417 Ki = 20 nM T84631 CT3BN9 10951324 Ki = 18 nM T84631 C2TBO9 10959252 Ki = 26000 nM T84631 C0B9VT 10960935 Ki = 1400 nM T84631 CB9KP4 10961420 Ki = 21 nM T84631 C6ZT5K 10961564 Ki = 1200 nM T84631 C8MSV2 10961726 Ki = 325 nM T84631 C9RTW1 10961857 Ki > 1200 nM T84631 CITU70 10962439 Ki > 75000 nM T84631 CCE31H 10963578 IC50 = 185 nM T84631 CJ29QP 10972004 Ki = 183 nM T84631 CH0VN7 10972370 IC50 > 30000 nM T84631 CFC7J3 10972388 Ki = 300 nM T84631 CT6Q7Z 10972928 Ki = 39 nM T84631 CIU42D 10973463 IC50 > 30000 nM T84631 C6HG4P 10974490 IC50 = 2700 nM T84631 CVT26S 10974535 IC50 = 540 nM T84631 CH41ZW 10974733 IC50 = 2400 nM T84631 CE0F1L 10983499 Ki > 1200 nM T84631 CPO91R 10983794 Ki = 13 nM T84631 CL9V7T 10984300 Ki = 18 nM T84631 CWVR40 10985371 IC50 = 2000 nM T84631 C9Y8LS 10991007 Ki = 6 nM T84631 CB79YS 10993022 Ki = 3327 nM T84631 C3RCS5 10994039 Ki = 900 nM T84631 CN0T4L 10994091 Ki = 690 nM T84631 CM5Y6J 10994432 IC50 > 30000 nM T84631 C4VA7K 10994660 IC50 > 30000 nM T84631 CZM0S7 10995244 Ki = 360 nM T84631 CT7L2Q 10996309 IC50 = 1000 nM T84631 C43SNO 11004109 Ki = 89 nM T84631 CF26JG 11004176 Ki = 280 nM T84631 CK3N5I 11004200 Ki = 620 nM T84631 CV86TU 11004465 Ki = 370 nM T84631 CP68KV 11004693 Ki = 460 nM T84631 C8AG4Z 11005226 IC50 > 30000 nM T84631 C12REQ 11005350 Ki = 918 nM T84631 CWHG91 11005419 Ki = 180 nM T84631 C0FG9E 11006294 Ki = 60 nM T84631 CC39SB 11009950 Ki = 125000 nM T84631 C3HW2I 11014107 Ki = 3300 nM T84631 CYZL25 11015002 Ki = 210 nM T84631 CFO15P 11015356 IC50 > 30000 nM T84631 CE7BX4 11015410 Ki = 1230 nM T84631 C56HDX 11015700 Ki > 5000 nM T84631 C5IS6E 11016482 Ki = 23 nM T84631 CV8O4G 11016622 Ki = 3 nM T84631 C49NMW 11022696 Ki = 5650 nM T84631 CM37HW 11025449 Ki = 1300 nM T84631 C71KSB 11026329 Ki > 1200 nM T84631 C4EX2J 11026555 Ki > 5000 nM T84631 CYKF85 11026584 Ki = 810 nM T84631 C21MKH 11026850 Ki = 140 nM T84631 CD4LJ1 11027118 IC50 > 30000 nM T84631 C46ZEX 11027375 Ki = 19 nM T84631 CI0VR4 11028729 Ki = 82 nM T84631 C2RG6V 11028969 IC50 = 180 nM T84631 CMQ65P 11035180 Ki = 2986 nM T84631 C3QG7H 11036285 Ki = 20 nM T84631 CV1F8Q 11036379 Ki = 170 nM T84631 C5KTL2 11037540 Ki = 89 nM T84631 CXO97Q 11037642 Ki = 25 nM T84631 CDGL91 11037810 Ki = 2043 nM T84631 C7PDA1 11037845 Ki = 17350 nM T84631 C9KL0E 11037866 Ki = 7030 nM T84631 C4LPB1 11039096 Ki > 5000 nM T84631 C7RM5W 11039881 IC50 = 210 nM T84631 C7P5EN 11039916 IC50 = 2180 nM T84631 C7VX2Y 11046972 Ki = 3200 nM T84631 CSQT80 11048143 Ki = 1118 nM T84631 CMBL62 11048452 Ki = 9 nM T84631 CA1U0X 11048482 Ki = 10000 nM T84631 CJL15S 11048586 Ki = 63 nM T84631 CF01BA 11049038 Ki = 19 nM T84631 C4SW1T 11049045 Ki = 1022 nM T84631 C4UY7P 11050903 IC50 = 770 nM T84631 CD9WJ8 11057540 Ki = 340 nM T84631 C2Y6VW 11057779 Ki = 14 nM T84631 CQ61ZR 11059085 IC50 > 30000 nM T84631 CJZ10A 11059370 Ki = 3000 nM T84631 C7IA8Y 11059381 Ki = 3804 nM T84631 CZ43QG 11059512 Ki = 1400 nM T84631 CX09AC 11059549 Ki > 5000 nM T84631 CH1OX5 11059588 Ki = 4 nM T84631 C8BC4U 11059598 Ki > 1200 nM T84631 CXW4P2 11059783 Ki = 160 nM T84631 C8L9KE 11059896 IC50 > 30000 nM T84631 CYG09F 11059945 Ki = 370 nM T84631 CRK76W 11060981 Ki = 140 nM T84631 CVGU32 11067332 Ki = 13000 nM T84631 C3HNB2 11068806 Ki = 78 nM T84631 CU02AK 11069944 Ki = 959 nM T84631 CJ4U7M 11069959 Ki = 5200 nM T84631 C7CX9Y 11070206 Ki = 128 nM T84631 C5D6CK 11070239 Ki = 77 nM T84631 CZY36H 11071021 Ki = 1628 nM T84631 CZU7P2 11071979 Ki = 94 nM T84631 C7YDH0 11072681 IC50 = 150 nM T84631 CDKX73 11080299 Ki = 263 nM T84631 CW3QV0 11080411 Ki = 2100 nM T84631 CZ5PW9 11080476 Ki = 308 nM T84631 CSE89U 11081058 Ki = 1219 nM T84631 CZ73WT 11081112 Ki = 3 nM T84631 C0FVC8 11082011 Ki = 61 nM T84631 CRIM63 11082881 Ki = 245 nM T84631 C2XYV1 11091496 Ki = 970 nM T84631 CB21LS 11092876 Ki = 1820 nM T84631 CXO16G 11092974 Ki = 14 nM T84631 CUX7H5 11098880 Ki = 7160 nM T84631 C0UP3R 11101386 Ki = 2032 nM T84631 C9CUO6 11102065 IC50 > 30000 nM T84631 C2XAM1 11102245 Ki = 650 nM T84631 CM1F6C 11102508 Ki = 2200 nM T84631 CY3M6F 11102509 Ki = 2400 nM T84631 C7DF0B 11102544 Ki = 193 nM T84631 C8R5EM 11102680 Ki = 476 nM T84631 CVB8L0 11102692 Ki = 37 nM T84631 C1U0NG 11102698 Ki = 841 nM T84631 C1GY8M 11102714 Ki = 1400 nM T84631 CU53EA 11104490 IC50 = 250 nM T84631 C41PZK 11112423 Ki = 64 nM T84631 C9KE6A 11112625 Ki = 210 nM T84631 C59EGY 11112713 Ki = 240 nM T84631 CI3N0C 11112769 Ki = 1360 nM T84631 CPD34Y 11112824 Ki = 48 nM T84631 CZV69J 11112866 Ki = 1200 nM T84631 CANW92 11112933 IC50 > 30000 nM T84631 CC37UH 11113237 Ki = 274 nM T84631 CAGC62 11113397 Ki = 304 nM T84631 CKL74M 11113517 Ki = 3 nM T84631 CS14TD 11113557 Ki = 318 nM T84631 CBY3A4 11113676 Ki > 5000 nM T84631 C30NPX 11113694 Ki = 2800 nM T84631 CEP79U 11122516 Ki > 5000 nM T84631 CDIS79 11122714 Ki = 1600 nM T84631 C03CFY 11122823 Ki > 5000 nM T84631 CALC18 11123099 Ki = 2000 nM T84631 CE4DH7 11123192 Ki = 173 nM T84631 CJBF29 11123629 Ki = 117 nM T84631 C39ATZ 11124077 Ki = 5000 nM T84631 CT50NB 11124237 Ki = 170 nM T84631 C47UEP 11125405 IC50 = 900 nM T84631 CD71SV 11125697 IC50 = 500 nM T84631 C0KYJ6 11133405 Ki = 1608 nM T84631 C39IZS 11134001 Ki = 4500 nM T84631 CT7S6O 11134002 Ki > 5000 nM T84631 CQ7X3J 11134090 Ki = 707 nM T84631 CY7E9X 11135514 Ki = 610 nM T84631 CD56CJ 11135734 Ki = 141 nM T84631 C0SG9J 11136398 IC50 = 250 nM T84631 C9KL8Y 11144992 Ki > 1200 nM T84631 CMX1S2 11146905 IC50 = 330 nM T84631 CWMD96 11146965 IC50 = 2770 nM T84631 C1NMK4 11146971 IC50 = 310 nM T84631 CS1K9H 11156015 Ki = 225200 nM T84631 C2TL3I 11156562 Ki = 110 nM T84631 CK3RG5 11157000 Ki = 2.9 nM T84631 CT2ML6 11157065 Ki = 10000 nM T84631 CJ4X7R 11158066 IC50 = 65000 nM T84631 C83DUK 11164311 IC50 = 3340 nM T84631 C5KG1A 11164549 Ki > 10000 nM T84631 CRD42J 11168063 Ki = 7.1 nM T84631 C3WKQ1 11168297 Ki = 2.8 nM T84631 CRG25K 11168660 IC50 = 190 nM T84631 C8KQY0 11168755 Ki = 10000 nM T84631 C58IYE 11169197 Ki = 17300 nM T84631 CIF5K2 11178928 Ki = 2 nM T84631 CZC46I 11179149 IC50 = 26 nM T84631 COM9K4 11179316 IC50 = 4300 nM T84631 CTM80Q 11179758 IC50 = 74 nM T84631 CEO0A3 11179888 Ki = 7 nM T84631 CU9K4E 11180045 IC50 = 22 nM T84631 C9X4JY 11181893 Ki = 0.37 nM T84631 CR0S7Z 11188883 Ki = 7800 nM T84631 CY70EN 11191165 IC50 > 10000 nM T84631 CB25UF 11191236 Ki = 1.1 nM T84631 C2RVF5 11191430 IC50 = 320 nM T84631 C68FEJ 11191721 IC50 = 105 nM T84631 CER29V 11197304 IC50 > 5000 nM T84631 CWA6L1 11202766 IC50 = 230 nM T84631 CAM0I3 11203305 Ki = 54 nM T84631 CJ6CW4 11203935 Ki = 38 nM T84631 C9J5HC 11212885 Ki = 87 nM T84631 CVG72J 11213445 Ki = 2221 nM T84631 CR5S8A 11214337 Ki = 2518 nM T84631 C9BY1M 11214717 Ki = 950 nM T84631 CO7H9G 11214939 Ki = 16590 nM T84631 CKH8E1 11215005 Ki = 71 nM T84631 C8BRJ1 11225386 Ki = 5.3 nM T84631 CSJW59 11226109 Ki = 7 nM T84631 CYQ3J1 11226153 Ki = 4327 nM T84631 C7MT4K 11226168 Ki = 5755 nM T84631 C7DJT1 11226460 Ki = 8 nM T84631 CP51FI 11226542 Ki = 1.7 nM T84631 CQZ7S2 11236581 Ki = 140 nM T84631 CVK0I4 11237021 IC50 = 1980 nM T84631 CLA93S 11237163 Ki = 0.67 nM T84631 CB29QS 11237358 Ki = 1540 nM T84631 CY8O2E 11237428 Ki = 7700 nM T84631 C37VTL 11238193 Ki = 62 nM T84631 CA3IS9 11248439 Ki = 2.8 nM T84631 CI0NE7 11248994 Ki = 9 nM T84631 CUP5C4 11249230 Ki = 1 nM T84631 C98HOZ 11249318 Ki = 1.8 nM T84631 C75IPG 11249648 Ki = 124 nM T84631 CE2JK3 11249816 Ki = 264 nM T84631 CHQ50D 11260319 IC50 = 420 nM T84631 CI9D8E 11260802 Ki = 10000 nM T84631 CN0EI2 11260937 Ki = 1051 nM T84631 CF0WU1 11261069 Ki = 4883 nM T84631 C7WIZ3 11261098 IC50 = 2900 nM T84631 C9MJA2 11271356 Ki = 2820 nM T84631 C2AFH8 11271916 IC50 = 230 nM T84631 CRDU42 11271947 Ki = 15 nM T84631 CYRO76 11272254 IC50 = 60 nM T84631 CW4OK6 11272980 Ki = 18 nM T84631 C92KFX 11273269 IC50 = 110 nM T84631 C73WSC 11273795 IC50 > 20000 nM T84631 CQP45I 11283566 Ki = 2 nM T84631 CZJ9C8 11283614 IC50 = 718 nM T84631 C91BDA 11284460 IC50 = 1900 nM T84631 CSH76U 11284767 Ki = 54600 nM T84631 CJ82SB 11294750 IC50 = 493 nM T84631 CO7LS5 11294802 Ki = 26 nM T84631 CEF02R 11294993 Ki = 0.53 nM T84631 CXQO17 11295553 Ki = 2574 nM T84631 C2WG5Z 11295972 Ki = 8 nM T84631 C3ZX2E 11295984 Ki = 810 nM T84631 CL79GU 11303092 IC50 = 4060 nM T84631 CTZ7X4 11306388 Ki = 2 nM T84631 CNCL81 11306615 Ki = 21 nM T84631 CA80VZ 11306712 Ki = 16 nM T84631 CL2GZ0 11306789 IC50 = 160 nM T84631 C71PYV 11307226 IC50 = 22 nM T84631 C72IDM 11307246 Ki = 47 nM T84631 C7L9MF 11307344 Ki = 421 nM T84631 C0TUI9 11307532 Ki = 0.54 nM T84631 CF9RM8 11307929 Ki = 17 nM T84631 CNUP65 11316684 Ki = 1.1 nM T84631 C5ZC1G 11317814 Ki = 2 nM T84631 C3L6GK 11318187 IC50 = 230 nM T84631 CP08JC 11318191 IC50 = 550 nM T84631 C7ZS2B 11320069 Ki = 0.7 nM T84631 CY87CQ 11329232 Ki = 5410 nM T84631 C14AWK 11329397 Ki = 1412 nM T84631 CTXB71 11329441 IC50 = 270 nM T84631 CUCB51 11329534 Ki = 3 nM T84631 C4K3SW 11329788 Ki = 3925 nM T84631 C3J7WN 11329826 IC50 = 255 nM T84631 CB46ZC 11329971 IC50 = 210 nM T84631 CVAI21 11330048 Ki = 3.6 nM T84631 CC6O0W 11340558 Ki = 8.1 nM T84631 CJI8G5 11340774 IC50 = 800 nM T84631 CSJZ70 11341303 Ki = 960 nM T84631 CW7E9F 11341378 Ki = 2184 nM T84631 C64EOX 11341794 Ki = 28 nM T84631 CR8NW9 11351302 Ki = 1.5 nM T84631 CK28PW 11351714 Ki = 173 nM T84631 CY9D3C 11352421 IC50 = 5.5 nM T84631 C12OTG 11352538 Ki = 20 nM T84631 C3FC4B 11352678 Ki = 17 nM T84631 CSIM71 11353123 Ki = 20 nM T84631 C1HON4 11353394 Ki = 153 nM T84631 C1V5ES 11363818 IC50 = 1350 nM T84631 CQ9BZ3 11363906 Ki = 42 nM T84631 CVA12Y 11363985 Ki = 3 nM T84631 CK51RW 11364032 Ki = 24 nM T84631 CT83NF 11364269 Ki = 22 nM T84631 C1ZGT7 11364310 Ki = 10000 nM T84631 CR04CN 11364346 Ki = 0.7 nM T84631 CY2HW5 11365859 Ki = 4.5 nM T84631 CBU78I 11373015 IC50 = 510 nM T84631 C4U9OQ 11374975 IC50 = 510 nM T84631 C52YOA 11375433 IC50 = 390 nM T84631 CDS70L 11375712 IC50 = 247 nM T84631 CUNB34 11377164 IC50 = 83 nM T84631 CJBD34 11386051 Ki = 2.6 nM T84631 CWUY06 11386385 Ki = 5 nM T84631 CB41UN 11386766 Ki = 1265 nM T84631 CIWL90 11386810 Ki = 10 nM T84631 COQH61 11387388 Ki = 55 nM T84631 C8URO7 11387451 Ki = 0.88 nM T84631 C6U5OI 11387989 Ki = 61 nM T84631 CDC76X 11396607 Ki = 9.5 nM T84631 CZ4EM5 11397605 Ki = 4.4 nM T84631 C5MYX8 11397764 Ki = 2.6 nM T84631 CV4I7J 11397824 IC50 = 6200 nM T84631 CVU08E 11397915 IC50 = 3.5 nM T84631 CU5H0T 11398145 IC50 = 270 nM T84631 C1MS0G 11398207 Ki = 6200 nM T84631 C2M1OW 11398411 Ki = 970 nM T84631 CM34VR 11398878 Ki = 10000 nM T84631 CR9Q3O 11399867 IC50 = 1400 nM T84631 C3O9MG 11408346 Ki = 4219 nM T84631 CS8TK0 11408450 Ki = 1.8 nM T84631 CR9Y7U 11408532 Ki = 4.7 nM T84631 C3DQ7J 11409073 IC50 = 120 nM T84631 C3KYM8 11409900 IC50 = 190 nM T84631 CPF6V4 11410761 Ki = 10000 nM T84631 C8WZ0P 11416498 Ki > 10000 nM T84631 CJI48N 11419907 Ki = 9345 nM T84631 CAI3Y6 11420126 Ki = 74 nM T84631 CODR29 11420832 Ki > 75000 nM T84631 CR9OZ8 11420936 Ki = 14 nM T84631 C8R5QT 11420982 Ki = 10000 nM T84631 CUHD35 11421628 Ki = 800 nM T84631 CTY4I2 11431806 Ki = 230 nM T84631 C9HIK8 11432017 Ki = 1128 nM T84631 C9UE5W 11432325 Ki = 5 nM T84631 CZ3C9N 11432971 Ki = 9 nM T84631 CH74DF 11433275 Ki = 835 nM T84631 CLH6X5 11433511 Ki = 1 nM T84631 CCPU80 11434124 Ki = 7.7 nM T84631 CN46CG 11441985 IC50 = 56 nM T84631 CW36NJ 11442160 Ki = 406 nM T84631 C9DQ6J 11443267 Ki = 34 nM T84631 CSI0R8 11443686 Ki = 3040 nM T84631 CNU51Z 11443953 Ki = 1484 nM T84631 CZ2YU6 11444061 Ki = 10000 nM T84631 CH7X6T 11444549 Ki = 10000 nM T84631 CIQH43 11445130 IC50 = 3600 nM T84631 CM7DK5 11445304 Ki = 0.16 nM T84631 C10PTA 11454249 Ki = 1 nM T84631 CFL61Z 11454667 Ki = 270 nM T84631 CB60QJ 11455408 Ki = 15 nM T84631 COC38U 11455413 Ki = 6217 nM T84631 C05LOJ 11455486 IC50 = 86 nM T84631 CG8H7N 11465140 IC50 = 5.5 nM T84631 CNF2M3 11465752 Ki = 650 nM T84631 CWC4B0 11465955 Ki = 3.7 nM T84631 C7B1LU 11466448 Ki = 10000 nM T84631 CYSI10 11466604 Ki = 13 nM T84631 CX31CK 11466687 Ki = 57 nM T84631 C89DVO 11466821 Ki = 1247 nM T84631 C8KJ1G 11466928 Ki = 110 nM T84631 C13CGX 11466988 Ki = 31 nM T84631 CU9LH8 11466995 IC50 = 400 nM T84631 C0T6CN 11467119 Ki = 600 nM T84631 CH4V9C 11468062 Ki = 0.1 nM T84631 CUF04L 11468141 Ki = 163 nM T84631 CJ6TL8 11468217 Ki = 0.52 nM T84631 C6P9OD 11477087 IC50 = 1300 nM T84631 CAC5N9 11477894 Ki = 2.3 nM T84631 CD31BU 11478099 IC50 = 5440 nM T84631 CLO07F 11478314 Ki = 10000 nM T84631 CU04WZ 11478333 Ki = 2.4 nM T84631 C85JCH 11478408 Ki = 130 nM T84631 C73GXV 11479028 Ki = 18 nM T84631 CVI82D 11479420 Ki = 0.09 nM T84631 CDKN64 11488503 Ki = 4.2 nM T84631 CGY6X5 11488924 Ki = 407 nM T84631 CB1PG7 11489024 IC50 = 640 nM T84631 CF15XY 11489042 IC50 = 920 nM T84631 C5DFC7 11489269 IC50 = 1200 nM T84631 CC5DO0 11489287 IC50 = 2200 nM T84631 CU2JO0 11489417 Ki = 463 nM T84631 C50FQZ 11489885 Ki > 200000 nM T84631 CI65TJ 11490312 IC50 = 80 nM T84631 C9R6LC 11496149 Ki = 4 nM T84631 C84NJM 11496686 IC50 = 3.6 nM T84631 CZ30GX 11497599 Ki = 5.5 nM T84631 C81ZHR 11503981 Ki = 0.33 nM T84631 CK34OX 11509611 Ki > 8180 nM T84631 CO1AY9 11509879 Ki = 223 nM T84631 CJZ09N 11512593 Ki = 5100 nM T84631 C28BMR 11513105 Ki = 4900 nM T84631 CLN0W3 11517577 IC50 = 1170 nM T84631 C1BV2R 11518043 IC50 = 197 nM T84631 C13UZL 11518307 Ki = 0.19 nM T84631 CLT1I0 11518907 Ki = 0.033 nM T84631 CKAE28 11519499 Ki = 3 nM T84631 CV6JF2 11523750 IC50 = 74 nM T84631 CO68MA 11524737 Ki > 8180 nM T84631 C0A6TY 11524901 IC50 = 2300 nM T84631 CKN8R7 11525275 IC50 = 1900 nM T84631 C20NQD 11525292 IC50 = 1.4 nM T84631 CRNU10 11534959 Ki = 4100 nM T84631 C9M6JZ 11538422 Ki = 2900 nM T84631 CUY97G 11539245 IC50 = 94 nM T84631 CD1A6T 11542037 Ki = 2800 nM T84631 CA8KD7 11542038 Ki = 1200 nM T84631 CKY49D 11546456 IC50 = 2000 nM T84631 CDS27O 11553603 IC50 = 40 nM T84631 CLQ1A9 11554212 IC50 = 8.5 nM T84631 CBP69L 11557024 Ki = 9500 nM T84631 CE4DV8 11561857 Ki = 5 nM T84631 CKJC51 11561914 Ki = 6 nM T84631 C2KM3Z 11562451 IC50 = 1 nM T84631 C3EMG1 11562571 IC50 = 2.3 nM T84631 CCG84F 11563457 Ki = 2300 nM T84631 CV46NL 11563632 Ki > 1000000 nM T84631 C4JLC8 11569203 IC50 = 0.4 nM T84631 CEAZ46 11569930 Ki = 66000 nM T84631 C3TJ7M 11570580 Ki = 1800 nM T84631 C6RHD8 11570700 Ki = 13000 nM T84631 C1DN2L 11570759 Ki = 80000 nM T84631 C9R6VJ 11575714 IC50 = 1260 nM T84631 C6FG8V 11577055 Ki = 76000 nM T84631 CIY34V 11577968 Ki = 8300 nM T84631 CJ38EP 11577970 Ki = 10500 nM T84631 C7MF9N 11578158 Ki = 3200 nM T84631 C6A0XP 11583256 IC50 = 2.5 nM T84631 C5W7FH 11583355 Ki = 5 nM T84631 C76BVQ 11583800 IC50 = 9.1 nM T84631 CTSK74 11584729 Ki = 21000 nM T84631 C96GNS 11585914 IC50 = 9500 nM T84631 C5W4SM 11590677 Ki = 0.3 nM T84631 C1RQ6P 11592130 Ki = 23000 nM T84631 CBC84M 11592593 Ki = 13000 nM T84631 C7ZS8L 11592600 Ki = 4600 nM T84631 C7QTY8 11606981 Ki = 2000 nM T84631 CU07NO 11607091 Ki = 17000 nM T84631 CC94FI 11612290 Ki = 0.028 nM T84631 CL9TZ2 11614477 Ki = 5000 nM T84631 C78TFB 11618984 IC50 = 290 nM T84631 CA56HC 11619782 IC50 = 1200 nM T84631 CB4O2Q 11621579 Ki = 2800 nM T84631 CD3R1E 11627899 Ki = 35000 nM T84631 CB9P0Q 11628768 Ki = 10000 nM T84631 CO3Q9N 11635973 Ki = 9000 nM T84631 CRX98P 11636026 Ki = 2800 nM T84631 C8N5CR 11638121 Ki = 1 nM T84631 CMC85Y 11641579 Ki = 3 nM T84631 CW10CL 11642802 Ki = 25000 nM T84631 C1O5ZV 11648797 Ki = 314000 nM T84631 CE3D4T 11650066 IC50 = 7.6 nM T84631 CZL5O6 11650704 Ki = 5.2 nM T84631 C7NG4M 11652744 Ki = 1 nM T84631 C2W5XF 11656797 Ki = 15000 nM T84631 C4SAR0 11657278 Ki = 1300 nM T84631 CVQ16C 11664107 Ki = 34000 nM T84631 CPZG49 11664334 Ki = 130000 nM T84631 CT9E0G 11664643 Ki = 2900 nM T84631 CWV87X 11671266 Ki = 15000 nM T84631 CE0A6N 11671776 Ki = 5300 nM T84631 C85GCY 11671956 Ki = 5800 nM T84631 C1IMQ2 11677338 Ki = 0.06 nM T84631 C1DHO6 11678360 Ki = 24000 nM T84631 C4IBO3 11678764 Ki = 2200 nM T84631 CJP9O1 11684611 Ki = 6390 nM T84631 C69YSR 11693028 Ki = 6300 nM T84631 CCQY30 11693049 Ki = 4000 nM T84631 CS27RX 11697174 Ki = 175 nM T84631 C0YO6U 11698686 Ki = 0.2 nM T84631 CPFW75 11699600 Ki = 13000 nM T84631 C3VS2H 11699903 Ki = 2300 nM T84631 CNV09Z 11699913 Ki = 1000 nM T84631 CI96PN 11704628 Ki = 124 nM T84631 C89KHJ 11707555 IC50 = 9600 nM T84631 CCVY81 11711363 IC50 = 4.2 nM T84631 CM57QZ 11718954 IC50 = 29 nM T84631 CKQ4O2 11721188 Ki = 56000 nM T84631 C4UB2X 11721375 Ki = 10000 nM T84631 C4M0XP 11725377 IC50 = 940 nM T84631 CJZA24 11729069 Ki = 2500 nM T84631 CL4CN3 11729890 Ki = 208 nM T84631 CS12RM 11730232 Ki = 45 nM T84631 CBJ4R6 11730277 Ki = 12000 nM T84631 CQ0ZP6 11730472 Ki > 1200 nM T84631 CL8HU6 11730709 IC50 > 30000 nM T84631 C7D8HR 11731179 Ki = 99 nM T84631 CN70PY 11732209 Ki = 1112 nM T84631 CW1U7K 11732650 Ki = 2190 nM T84631 C0VO1S 11732813 Ki = 191 nM T84631 C8K1ZJ 11733007 Ki = 720 nM T84631 C7LW3O 11734113 Ki = 100 nM T84631 CNZ04Q 11740591 Ki = 1400 nM T84631 CR53AD 11742672 Ki = 3 nM T84631 C8QZK0 11743193 Ki = 80 nM T84631 CO12HL 11743369 Ki = 495 nM T84631 C5VN3J 11744466 Ki = 2.7 nM T84631 CM95SZ 11744578 IC50 = 1 nM T84631 C7DHE6 11752478 Ki = 6515 nM T84631 C27LUA 11752612 IC50 = 160 nM T84631 CCBH57 11752638 Ki = 306 nM T84631 C5C3BR 11752747 Ki = 24 nM T84631 CX18BY 11752965 Ki = 4.2 nM T84631 CQ81KJ 11753784 IC50 = 122 nM T84631 CP3FI1 11753847 Ki > 15000 nM T84631 C1LPF4 11754261 IC50 = 14 nM T84631 CV62MN 11754356 IC50 = 58 nM T84631 CZ2W6F 11754502 Ki = 3300 nM T84631 C8GJO7 11754872 IC50 = 9.3 nM T84631 CNPW05 11755188 Ki = 0.7 nM T84631 CUMO51 11756555 IC50 = 58 nM T84631 CTOM97 11756558 Ki = 169 nM T84631 C9XAJ5 11756561 Ki = 0.12 nM T84631 CS0JR2 11756961 Ki = 0.83 nM T84631 CMR6A0 11758260 Ki > 8000 nM T84631 C7P4CG 11758475 Ki = 5900 nM T84631 CMD7Z1 11760447 Ki = 5000 nM T84631 CG82LK 11761121 Ki = 1400 nM T84631 CZ7QI3 11761613 Ki = 125 nM T84631 C82ULR 11761706 Ki = 700 nM T84631 CDLZ28 11761967 Ki = 44 nM T84631 CJVR18 11762113 Ki = 1300 nM T84631 CHQ58K 11762202 Ki = 131 nM T84631 C0C9KI 11762303 Ki > 1200 nM T84631 CL53HV 11762323 Ki = 4 nM T84631 CZ91LI 11762766 Ki > 75000 nM T84631 COM9B5 11763170 IC50 > 30000 nM T84631 CWR03Q 11766372 IC50 = 210 nM T84631 CR2E9T 11782463 Ki = 43 nM T84631 C9LC5W 11784323 Ki = 5000 nM T84631 CRH1M7 11784791 Ki = 0.7 nM T84631 C7M3TO 11785263 Ki = 3 nM T84631 CL7QS3 11785424 Ki = 4035 nM T84631 C85MUK 11785772 Ki = 1378 nM T84631 C1EQX3 11785872 Ki = 167 nM T84631 CN3IG5 11785929 Ki = 10 nM T84631 CK4CH2 11786303 Ki = 10 nM T84631 CU9RW5 11792439 Ki = 2700 nM T84631 C8LD7W 11793807 Ki > 5000 nM T84631 CAGC25 11795137 Ki = 160 nM T84631 CZ62LI 11796080 Ki = 960 nM T84631 CW6DG1 11796805 Ki = 1600 nM T84631 CF1S2R 11796942 Ki > 5000 nM T84631 CIS51A 11797515 Ki = 94000 nM T84631 CZM62X 11797951 Ki = 110 nM T84631 CNO67W 11798089 Ki = 5200 nM T84631 CH2Z1N 11798267 Ki = 89 nM T84631 CK8MI3 11798429 Ki = 420000 nM T84631 CK31IT 11800766 Ki = 19 nM T84631 CL6Z3G 11801417 Ki = 16000 nM T84631 C68VNG 11801427 Ki = 210 nM T84631 CL01GT 11801580 Ki = 7.2 nM T84631 CVZ82O 11801725 Ki = 200 nM T84631 CFP36D 11802531 Ki = 13 nM T84631 CY46UZ 11802721 Ki = 5.3 nM T84631 C09WKB 11813114 Ki = 2400 nM T84631 C9VW2P 11813305 Ki = 8 nM T84631 C6W0VT 11813820 Ki = 66 nM T84631 C47BFQ 11813993 Ki = 76 nM T84631 C1Y5NB 11814014 Ki = 144 nM T84631 CUN1S4 11814234 Ki = 134 nM T84631 C8INH6 11814686 IC50 = 3140 nM T84631 C7JO4I 11823405 Ki = 8800 nM T84631 C98ZOR 11824040 Ki = 19000 nM T84631 CYX74A 11824584 Ki = 5200 nM T84631 CCT84E 11825785 Ki > 5000 nM T84631 CEYP62 11826299 Ki = 51 nM T84631 C79MQD 11826825 IC50 > 30000 nM T84631 C3EFY7 11826875 Ki = 61 nM T84631 C93TLO 11827247 Ki = 26 nM T84631 C9R2OA 11828043 Ki = 103 nM T84631 C61GPA 11828451 IC50 = 2100 nM T84631 CW6E7I 11828640 IC50 = 210 nM T84631 C4DTE8 11849112 Ki = 1 nM T84631 CY8T0B 11950081 Ki = 0.6 nM T84631 CQ74TC 11950083 Ki = 1 nM T84631 CN27JS 11950249 Ki = 1 nM T84631 CGY83S 11950253 Ki = 10 nM T84631 C6XW2E 11950427 Ki = 8 nM T84631 CRD0A6 11950428 Ki = 15 nM T84631 CTJ3A8 11950431 Ki = 1.3 nM T84631 CXH68R 11950432 Ki = 0.6 nM T84631 C9PV4Y 11950602 Ki = 2 nM T84631 CYX53O 11950605 Ki = 2 nM T84631 C86SCE 11950606 Ki = 1 nM T84631 CTZ4B6 11956166 Ki = 100 nM T84631 C6XRH4 11966394 Ki = 40 nM T84631 C5SEB3 11967063 IC50 = 1800 nM T84631 CTB2C9 11967128 IC50 = 380 nM T84631 CS92GP 11979006 Ki = 10 nM T84631 C12IZN 11979007 Ki = 3 nM T84631 C34NUJ 11979125 Ki = 10 nM T84631 CE04WI 11979126 Ki = 22 nM T84631 C69HNO 11984565 Ki = 7200 nM T84631 CPR4I1 12047383 Ki = 87000 nM T84631 C5U0FJ 12047384 Ki = 87000 nM T84631 C5FU3H 12047385 Ki = 45000 nM T84631 CX98PQ 12082573 IC50 = 500 nM T84631 CT7IR8 12110710 IC50 > 100000 nM T84631 CLJ15H 12222233 Ki = 6.8 nM T84631 C1TK9C 12972260 IC50 = 106 nM T84631 C1IT4G 12972261 IC50 = 62.6 nM T84631 C84CJL 12986348 IC50 = 260 nM T84631 CYN6H0 12988920 Ki = 0.72 nM T84631 CO5Z4Y 12989060 Ki = 0.29 nM T84631 CQ8OU1 13755335 Ki = 1800 nM T84631 C45LTS 13755337 Ki = 1300 nM T84631 C60TVD 15392306 IC50 = 6 nM T84631 C7ZV8R 15392323 IC50 = 6 nM T84631 C3HYW7 15431805 IC50 > 2500 nM T84631 CZBD56 15435386 Ki = 94 nM T84631 C9KJ5Y 15461560 Ki = 0.33 nM T84631 CM2RN1 15461564 Ki = 0.015 nM T84631 C5CQ6R 15463576 Ki = 3.4 nM T84631 CCN18Q 15463577 Ki = 13 nM T84631 CZ4L6O 15463578 Ki = 400 nM T84631 CF9H3Z 15463579 Ki = 460 nM T84631 CY2S1U 15463580 Ki = 12 nM T84631 CQTF26 15463581 Ki = 26 nM T84631 CX5S1Z 15511974 Ki = 2.1 nM T84631 CW2QY0 15515689 IC50 = 4100 nM T84631 CG9Q0P 15515690 IC50 = 2500 nM T84631 C54SUM 15515691 IC50 = 16000 nM T84631 C60JFG 15521694 Ki = 1450 nM T84631 CP63GF 15534822 IC50 > 2500 nM T84631 CPJT95 15545832 Ki = 180 nM T84631 CKQ8M6 15546794 Ki = 6 nM T84631 CI6G0C 15736732 IC50 = 2500 nM T84631 CL9T7Y 15870100 Ki = 2100 nM T84631 CB3T9P 15870101 Ki = 400 nM T84631 C9EH2Y 15887336 IC50 = 230 nM T84631 C6VZ1N 15942655 Ki = 125000 nM T84631 CA86KZ 15947513 Ki = 8100 nM T84631 CU0O5N 15947601 Ki = 3900 nM T84631 CQ3RF8 15947602 Ki = 1800 nM T84631 CS8HY6 15947811 Ki = 4100 nM T84631 CCMQ45 15947923 Ki = 7600 nM T84631 CUGI75 15947926 Ki = 6200 nM T84631 CSV70B 15948627 Ki = 7200 nM T84631 C7VH6K 15950345 Ki = 0.16 nM T84631 C4EW6F 15965462 IC50 = 4 nM T84631 CMYR94 15976119 Ki = 5077 nM T84631 CLP2D3 16004672 Ki = 0.033 nM T84631 CX7KR1 16040261 Ki = 534 nM T84631 CA8Y1K 16046152 Ki = 0.27 nM T84631 CNBJ60 16046153 Ki = 0.37 nM T84631 CC7Y0D 16066741 IC50 > 200000 nM T84631 C3EUJ6 16086336 IC50 = 33500 nM T84631 CDSM46 16098887 IC50 = 14000 nM T84631 CFK98M 16098895 IC50 = 1700 nM T84631 C6BQ0G 16098896 IC50 > 200000 nM T84631 C1ZXL4 16098897 IC50 = 8500 nM T84631 CP6Y7Q 16098898 IC50 = 22000 nM T84631 C3J6LO 16098899 IC50 > 200000 nM T84631 CQ4YJ8 16098900 IC50 = 15000 nM T84631 CDL2X5 16098901 IC50 = 13000 nM T84631 C53ZXO 16098902 IC50 > 20000 nM T84631 CUJ5A9 16098903 IC50 > 20000 nM T84631 CZ3WM4 16098905 IC50 > 200000 nM T84631 CVN8Y1 16098906 IC50 = 2700 nM T84631 CTY5W9 16098907 IC50 = 14900 nM T84631 C53YRO 16098910 IC50 = 1600 nM T84631 C91CQM 16098911 IC50 = 250 nM T84631 C0W5NR 16098912 IC50 = 1600 nM T84631 CS21OE 16098913 IC50 = 2100 nM T84631 CO08FM 16112849 Ki = 1 nM T84631 CTW28E 16124699 Ki = 109 nM T84631 CSG06K 16124700 Ki = 165 nM T84631 CO69AB 16124701 Ki = 163 nM T84631 C91VBY 16124702 Ki = 2898 nM T84631 C41KQS 16124703 Ki > 15800 nM T84631 CP82YG 16124704 Ki = 285 nM T84631 CY3F2H 16124761 Ki = 4160 nM T84631 CM3Q6R 16124762 Ki = 112 nM T84631 CPD7L0 16124763 Ki = 170 nM T84631 CA53KN 16124764 Ki = 5 nM T84631 CX2BE1 16125613 Ki = 314 nM T84631 CM3P5C 16125614 Ki = 3670 nM T84631 C6E7RC 16125615 Ki = 3225 nM T84631 C8SNI9 16125616 Ki = 782 nM T84631 CBH64D 16125617 Ki = 1200 nM T84631 CIQ7S3 16125671 Ki = 2 nM T84631 CU5YJ0 16125672 Ki = 24 nM T84631 CJ7E2X 16204383 IC50 = 1.2 nM T84631 CL7Z6K 16215018 IC50 = 3.9 nM T84631 CN6CJ2 16220264 IC50 = 6470 nM T84631 CZ7FS4 16284785 IC50 > 200000 nM T84631 C56TPZ 16285203 IC50 > 200000 nM T84631 C1KZB9 16289649 IC50 > 200000 nM T84631 CQ0EK7 16660960 IC50 = 2.1 nM T84631 CX4UT5 16660962 IC50 = 37 nM T84631 CL2W9Q 16660964 IC50 = 5.7 nM T84631 CG2Q8U 16660966 IC50 = 3.3 nM T84631 CX36RF 16660968 IC50 = 6.5 nM T84631 C27COL 16661109 IC50 = 0.43 nM T84631 CPK67M 16664096 Ki = 0.35 nM T84631 CU28CE 16718713 IC50 = 30000 nM T84631 CC20PS 16718760 IC50 = 250000 nM T84631 CCKO80 16718762 IC50 = 27000 nM T84631 CTZ74D 16718807 IC50 > 250000 nM T84631 C37MRI 16718808 IC50 > 10000 nM T84631 CUL0B3 16720561 Ki = 15.9 nM T84631 CJL72U 16731819 Ki = 0.43 nM T84631 C05JSB 16731821 Ki = 0.16 nM T84631 C6SN2Q 16731823 Ki = 0.36 nM T84631 CG49VM 16731824 Ki = 1 nM T84631 C8ZFY6 16731827 Ki = 0.4 nM T84631 CN60KL 16731975 Ki = 1.4 nM T84631 CB01OR 16731976 Ki = 0.22 nM T84631 C7MR9E 16731977 Ki = 1.4 nM T84631 CF4V3D 16731978 Ki = 0.52 nM T84631 CS2QJ8 16731979 Ki = 2.2 nM T84631 CYB1E0 16731980 Ki = 0.24 nM T84631 CD64LP 16732121 Ki = 0.18 nM T84631 CWU9D7 16732123 Ki = 0.4 nM T84631 CH2U5Z 16732125 Ki = 0.71 nM T84631 CSB43R 16732126 Ki = 0.26 nM T84631 CK74UL 16732127 Ki = 0.024 nM T84631 C4A1RO 16732128 Ki = 0.019 nM T84631 C9BD4C 16732263 Ki = 0.045 nM T84631 CZ3M6S 16732265 Ki = 0.026 nM T84631 C3DW7C 16732266 Ki = 0.02 nM T84631 CBO97E 16732268 Ki = 0.05 nM T84631 C7QBR0 16732402 Ki = 0.036 nM T84631 C6RPF4 16732404 Ki = 0.022 nM T84631 CN3D9T 16732406 Ki = 0.012 nM T84631 C1HFQ6 16732407 Ki = 2.2 nM T84631 CGC0Q2 16732555 Ki = 0.12 nM T84631 C7SUK0 16732557 Ki = 0.26 nM T84631 CT4K0V 16732559 Ki = 0.12 nM T84631 CKAZ40 16732560 Ki = 0.031 nM T84631 CKN73Z 16732562 Ki = 0.012 nM T84631 CLF90N 16732707 Ki = 0.026 nM T84631 CR3K2E 16732708 Ki = 0.024 nM T84631 C2EOR6 16732711 Ki = 0.004 nM T84631 CPK8Z7 16732713 Ki <= 0.01 nM T84631 CUHT92 16732866 Ki <= 0.01 nM T84631 C07OPV 16732868 Ki <= 0.01 nM T84631 C3Y2HE 16732871 Ki = 0.004 nM T84631 C47UEZ 16732873 Ki <= 0.01 nM T84631 CL4EW1 16733006 Ki = 0.004 nM T84631 CNYA03 16733007 Ki <= 0.01 nM T84631 C7XU2R 16733008 Ki <= 0.01 nM T84631 CRBI26 16733010 Ki = 0.022 nM T84631 CUEL18 16733012 Ki <= 0.01 nM T84631 C6OK0W 16733013 Ki = 0.006 nM T84631 C0G7KW 16733150 Ki = 0.02 nM T84631 C54HKA 16734339 Ki = 1.3 nM T84631 CJ3MX8 16734340 Ki = 0.8 nM T84631 C08JWR 16734545 Ki = 0.8 nM T84631 CF8S7J 16734546 Ki = 0.8 nM T84631 C7CSO3 16741235 IC50 = 0.16 nM T84631 COZ62I 16748993 IC50 = 0.38 nM T84631 CYDU97 16749087 IC50 = 18 nM T84631 CJG13M 17756142 IC50 = 4.6 nM T84631 C2K9GC 17788740 Ki = 170 nM T84631 CVB82P 17809181 IC50 = 880 nM T84631 CB6R1Z 17809213 IC50 = 6.63 nM T84631 C9PVW1 17822583 Ki = 2100 nM T84631 CF4K6R 17843517 IC50 = 123 nM T84631 C2IEC4 17851729 IC50 = 120 nM T84631 CA91IM 17851931 IC50 = 110 nM T84631 C16XHL 17852016 IC50 = 63 nM T84631 C72GHY 17852042 IC50 = 79 nM T84631 C5RSD3 18318130 Ki = 0.17 nM T84631 CL13IP 18318139 Ki = 0.56 nM T84631 C3P0VK 18318146 Ki = 6.8 nM T84631 COJ9F3 18318187 Ki = 0.55 nM T84631 C1S3MX 18318188 Ki = 0.88 nM T84631 CGNJ35 18318198 Ki = 7.5 nM T84631 CE7RZ4 18318201 Ki = 4.1 nM T84631 CBS40I 18318220 Ki = 0.27 nM T84631 COC54Y 18327622 Ki = 250000 nM T84631 CI5J3Y 18376546 Ki = 15 nM T84631 CMU9A3 18376555 Ki = 470 nM T84631 CFQE53 18376558 Ki = 26 nM T84631 CLUC36 18376562 Ki = 6.2 nM T84631 C76KJP 18376565 Ki = 54 nM T84631 CC94AD 18376598 Ki = 3.7 nM T84631 CJ7K3O 18376605 Ki = 10 nM T84631 C1UT4K 18376606 Ki = 1.6 nM T84631 CU98XE 18376618 Ki = 1.9 nM T84631 CCH92J 18376625 Ki = 34 nM T84631 C25PXL 18376627 Ki = 11 nM T84631 CL4UC9 18376641 Ki = 0.005 nM T84631 C4TCP6 18376642 Ki = 0.6 nM T84631 C0D1EH 18376656 Ki = 12 nM T84631 CN8CI1 18376659 Ki = 6 nM T84631 CTA57Y 18376663 Ki = 10 nM T84631 CHO4P2 18376665 Ki = 14 nM T84631 CPGX36 18376669 Ki = 0.8 nM T84631 CG0N9Q 18376671 Ki = 25 nM T84631 CU7V4F 18376679 Ki = 12 nM T84631 CIJG48 18376696 Ki = 2 nM T84631 C27NVA 18376714 Ki = 3.5 nM T84631 CR1C3F 18376717 Ki = 19 nM T84631 CSJZ89 18376719 Ki = 0.52 nM T84631 CUE92D 18376730 Ki = 73 nM T84631 CPT6W5 18376743 Ki = 58 nM T84631 CZ7HJ6 18376748 Ki = 24 nM T84631 CXW37R 18376768 Ki = 130 nM T84631 CBO4I0 18376780 Ki = 4.8 nM T84631 C7JF8K 18376782 Ki = 5.9 nM T84631 C86WAR 18376800 Ki = 2.3 nM T84631 CUZ8V3 18376816 Ki = 5 nM T84631 CAQ7X0 18376821 Ki = 590 nM T84631 C7Y8FD 18376826 Ki = 9.5 nM T84631 CRA3Y5 18376827 Ki = 7.2 nM T84631 C4I9XE 18376832 Ki = 0.45 nM T84631 C0S9XW 18376837 Ki = 24 nM T84631 CG98XS 18376838 Ki = 7.2 nM T84631 C4JE8S 18376839 Ki = 0.8 nM T84631 CN1ZX0 18376843 Ki = 2.1 nM T84631 C8YF1V 18376848 Ki = 16 nM T84631 CS79AF 18376858 Ki = 1.8 nM T84631 C9FDM4 18376865 Ki = 100 nM T84631 CUIC43 18376871 Ki = 2.1 nM T84631 CJL9E5 18376880 Ki = 1.4 nM T84631 C8KTW9 18376881 Ki = 22 nM T84631 C63EFY 18376882 Ki = 1.4 nM T84631 CE2BH4 18376888 Ki = 5.6 nM T84631 CE43LC 18376891 Ki = 21 nM T84631 C9V3HX 18376897 Ki = 18 nM T84631 C1ZKY8 18376901 Ki = 0.95 nM T84631 CH8R6S 18376905 Ki = 0.38 nM T84631 CUJP51 18376916 Ki = 260 nM T84631 CLE27U 18376919 Ki = 7.5 nM T84631 C3EN2U 18376921 Ki = 4.6 nM T84631 CM6NT1 18376930 Ki = 2.7 nM T84631 CG8Y0C 18376939 Ki = 5.2 nM T84631 C1SZ9Q 18376940 Ki = 210 nM T84631 CWG72T 18376950 Ki = 26 nM T84631 CV3ZE2 18376959 Ki = 14 nM T84631 CWI0E3 18376970 Ki = 2.2 nM T84631 C1OM7T 18376973 Ki = 0.3 nM T84631 C1T3VP 18376976 Ki = 1.6 nM T84631 C7SO8U 18376989 Ki = 150 nM T84631 CF0GR6 18376995 Ki = 7 nM T84631 CN2JE5 18376999 Ki = 30 nM T84631 CC9ZE2 18377002 Ki = 20 nM T84631 C53XHD 18377003 Ki = 1.7 nM T84631 C94LUS 18377010 Ki = 18 nM T84631 C79ZIE 18377020 Ki = 16 nM T84631 C3FYR1 18377031 Ki = 22 nM T84631 CI5U7D 18377033 Ki = 7 nM T84631 CEH2K1 18377041 Ki = 160 nM T84631 CX8RE3 18377048 Ki = 0.82 nM T84631 CN87FW 18474271 Ki = 2700 nM T84631 C3V9EC 18549309 Ki = 0.009 nM T84631 C63ILO 18549509 Ki = 0.09 nM T84631 C09CBT 18675029 IC50 = 26000 nM T84631 C0OPG9 18675052 IC50 = 5600 nM T84631 CRE8M4 18675059 IC50 = 27000 nM T84631 C9NB0Z 18675062 IC50 = 12 nM T84631 C09KIY 18675079 IC50 = 48 nM T84631 C29WYS 18675086 IC50 = 3 nM T84631 CR6I5L 18675103 IC50 = 16000 nM T84631 CLZ97R 18675188 IC50 = 7900 nM T84631 CFU8B9 18675209 IC50 = 66000 nM T84631 C17EDK 18675223 IC50 = 4900 nM T84631 C9NFX4 18675228 IC50 = 34000 nM T84631 CK6U1I 18675238 IC50 = 1600 nM T84631 CN0LW2 18675252 IC50 = 840 nM T84631 CM5VX3 18675291 IC50 = 23000 nM T84631 CD9UE4 18675298 IC50 = 68 nM T84631 CB01HJ 18675385 IC50 = 17000 nM T84631 CV5EG7 18727564 IC50 = 6 nM T84631 CWS58B 18727568 IC50 = 19 nM T84631 C2P5HW 18727569 IC50 = 1.2 nM T84631 C8ZP2O 18727570 IC50 = 1.5 nM T84631 C91FXK 18727571 IC50 = 16 nM T84631 COB7U9 18727572 IC50 = 12 nM T84631 CU3G4Q 18727574 IC50 = 4.8 nM T84631 CS8Y6P 18727576 IC50 = 10 nM T84631 C43RUO 18727577 IC50 = 5.4 nM T84631 CF4W5D 18727604 IC50 = 4 nM T84631 CB0IQ4 18727607 IC50 = 10 nM T84631 C6QZL7 18727622 IC50 = 1.2 nM T84631 CK2N1A 18727717 IC50 = 67 nM T84631 CNIB76 18727776 IC50 = 7.7 nM T84631 C9HXV5 18727777 IC50 = 370 nM T84631 C8AXM2 18727805 IC50 = 0.7 nM T84631 C31ZAL 18727831 IC50 = 15 nM T84631 CJY67O 18727833 IC50 = 2 nM T84631 C02HEA 18727834 IC50 = 15 nM T84631 CJSL38 18727836 Ki = 0.3 nM T84631 C8AMY9 18727838 IC50 = 7 nM T84631 CDO92V 18727840 IC50 = 2 nM T84631 CY8AC3 18727841 IC50 = 140 nM T84631 CB68ZV 18727844 IC50 = 0.6 nM T84631 C2M7ZO 18727846 IC50 = 0.6 nM T84631 C1IL8E 18727847 IC50 = 1.3 nM T84631 CD02TK 18727852 IC50 = 17 nM T84631 C1JMX5 18727855 IC50 = 16 nM T84631 CP7HL9 18727867 IC50 = 0.5 nM T84631 CQI72L 18727923 IC50 = 6060 nM T84631 CJM5I3 18727924 IC50 = 1810 nM T84631 C8GR2Q 18727965 IC50 = 78 nM T84631 CD51CF 18727967 IC50 = 714 nM T84631 CC0U9I 18727969 IC50 = 23 nM T84631 CL4B1V 18728102 IC50 = 226 nM T84631 C24ZCT 18728106 IC50 = 316 nM T84631 CKX4D1 18728109 IC50 = 7 nM T84631 CZ0XE6 18728123 IC50 = 0.7 nM T84631 C4DPW0 18728129 IC50 = 38 nM T84631 C0V4HL 18728139 IC50 = 26 nM T84631 C9OGD1 18728140 IC50 = 23 nM T84631 CJ4WA9 18728144 IC50 = 2 nM T84631 CE0ZU2 18728158 IC50 = 18 nM T84631 CNUR53 18800583 Ki = 400 nM T84631 C5MR0U 20585828 IC50 = 20 nM T84631 C7P4UB 20585829 IC50 = 10 nM T84631 CO2JG4 20595081 IC50 = 45 nM T84631 CGJN85 20595087 IC50 = 46 nM T84631 C9MN8Y 20595088 IC50 = 36 nM T84631 CM7BH1 20595091 IC50 = 24 nM T84631 CCH5N1 20595225 IC50 = 545 nM T84631 C70TFO 20595245 IC50 = 110 nM T84631 CX68HR 20595247 IC50 = 31 nM T84631 CX9YN6 20595251 Ki = 3.9 nM T84631 CKYA19 20595257 IC50 = 14 nM T84631 C2ID8R 20595260 Ki = 1.7 nM T84631 CH3D0Y 20595264 IC50 = 134 nM T84631 C8DXS5 20595268 IC50 = 28 nM T84631 C1HAM4 20595273 IC50 = 15 nM T84631 CM78XE 20595304 IC50 = 777 nM T84631 C10EGW 20595308 IC50 = 50 nM T84631 C0A9HN 20595310 IC50 = 50 nM T84631 CUS20T 20595326 IC50 = 16 nM T84631 CMT46A 20595328 Ki = 3.9 nM T84631 C9U2QS 20595336 IC50 = 18 nM T84631 C43UDK 20608737 IC50 > 30000 nM T84631 CW3I9O 20608738 IC50 > 30000 nM T84631 C4UZO0 20608741 IC50 > 30000 nM T84631 C9Z2VH 20608755 IC50 > 30000 nM T84631 C3OF2S 20608756 IC50 > 30000 nM T84631 CMX4Q6 20608776 IC50 > 30000 nM T84631 CXH09O 20631502 IC50 = 0.01 nM T84631 C2YDK5 20641721 IC50 = 4 nM T84631 CT7I1B 20641743 IC50 = 13 nM T84631 C7LHE8 20641745 Ki = 2.7 nM T84631 CTY8G2 20707887 Ki = 1.2 nM T84631 C0BKY3 20707927 IC50 = 2700 nM T84631 CB0X8I 20707929 IC50 = 650 nM T84631 C2BM9Q 20708041 IC50 = 1200 nM T84631 C7LX8J 20708044 IC50 = 1100 nM T84631 C0FRB4 20708055 IC50 = 60 nM T84631 CLM02X 20708056 IC50 = 380 nM T84631 C74LUP 20708058 IC50 = 50 nM T84631 CI6ZK4 20708066 IC50 = 180 nM T84631 CC3I4M 20708069 IC50 = 110 nM T84631 CJL5M6 20708073 IC50 = 360 nM T84631 CS57OI 20708074 IC50 = 890 nM T84631 CRK8N0 20708078 IC50 = 120 nM T84631 CC50OV 20708079 IC50 = 90 nM T84631 CK2V5A 20708094 IC50 = 700 nM T84631 CC7OB1 20708098 IC50 = 790 nM T84631 C6DN0A 20708099 IC50 = 160 nM T84631 C7JMO0 20708106 IC50 = 110 nM T84631 CR18VG 20708107 IC50 = 60 nM T84631 C02MHB 20708108 IC50 = 240 nM T84631 CL13GC 20708219 IC50 = 540 nM T84631 CWH2Z7 20747446 IC50 = 31 nM T84631 CXA98P 20747457 IC50 = 21 nM T84631 CV6KT1 20747459 IC50 = 61 nM T84631 CLZ5O4 20747496 IC50 = 93 nM T84631 CD2JP6 20747497 IC50 = 10 nM T84631 C2F4CK 20747503 IC50 = 256 nM T84631 C4CL5Y 20751605 IC50 = 64 nM T84631 CZ6KH9 20760195 Ki = 0.74 nM T84631 CH9J6I 20760215 Ki = 0.6 nM T84631 C7P9YE 20760216 Ki = 0.6 nM T84631 CR05LA 20760219 Ki = 3.6 nM T84631 C6ZUX8 20760222 Ki = 1.6 nM T84631 CMT78G 20760223 Ki = 3.8 nM T84631 CFY3L6 20801005 Ki = 474 nM T84631 C6IC3V 20801009 Ki = 73 nM T84631 C1DBA6 20801019 Ki = 57 nM T84631 CS29FI 20801029 Ki = 2230 nM T84631 CW0KR1 20801030 Ki = 400 nM T84631 CDIB13 20801031 Ki = 3 nM T84631 C65FLV 20801045 Ki = 654 nM T84631 C02ZCV 20801048 Ki = 9010 nM T84631 CTF5N7 20801076 Ki = 2500 nM T84631 CXQ3N0 20801082 Ki = 2100 nM T84631 CXR5A9 20801095 Ki = 810 nM T84631 C9RG0H 20801097 Ki = 4 nM T84631 CMI8H7 20801110 Ki = 220 nM T84631 CT7NZ2 20801115 Ki = 131 nM T84631 CUKR42 20801117 Ki = 64 nM T84631 C8KYF3 20801119 Ki = 106 nM T84631 CFJ13A 20801120 Ki = 71 nM T84631 CIM9C3 20801121 Ki = 27 nM T84631 CZW87C 20801125 Ki = 142 nM T84631 CB84ZQ 20801132 Ki = 20 nM T84631 CG51FK 20801137 Ki = 161 nM T84631 CC1Y0R 20801139 Ki = 40 nM T84631 CCO9S7 20801141 Ki = 125 nM T84631 C4V8ZR 20801142 Ki = 64 nM T84631 CCY5O7 20801143 Ki = 95 nM T84631 CY39JK 20801144 Ki = 95 nM T84631 COAC01 20801159 Ki = 15 nM T84631 CS3HB4 20801160 Ki = 40 nM T84631 CVSI76 20801207 Ki = 763 nM T84631 CCZJ48 20801208 Ki = 1075 nM T84631 CVNJ41 20801210 Ki > 10000 nM T84631 C3QBC1 20801212 Ki = 2480 nM T84631 CGD57F 20802932 IC50 > 30000 nM T84631 CO2FM4 20802944 IC50 > 30000 nM T84631 C1P0WC 20802959 IC50 > 30000 nM T84631 CBL6N1 20802966 IC50 > 30000 nM T84631 C27ZJT 20802995 IC50 > 100000 nM T84631 C3B4MA 20824147 IC50 = 8 nM T84631 C5ACM1 20843251 IC50 = 55000 nM T84631 C3RTJ2 20872059 Ki = 0.36 nM T84631 CG0RD2 21071205 Ki = 0.13 nM T84631 C95DUQ 21071251 Ki = 2.4 nM T84631 CR6C2I 21218691 Ki = 270 nM T84631 CS5L2M 21218709 Ki = 117 nM T84631 CEQ6B2 21218732 Ki = 20 nM T84631 C79ZNM 21218751 Ki = 143 nM T84631 CLT36V 21250176 IC50 = 500 nM T84631 CRYB96 21250293 IC50 = 400 nM T84631 C0ECB5 21250297 IC50 > 100000 nM T84631 CLV49W 21250386 IC50 = 9200 nM T84631 CN2YE9 21250416 IC50 = 46000 nM T84631 CRD4V1 21250427 IC50 = 1400 nM T84631 C3T5SA 21250434 IC50 = 31000 nM T84631 C9H7ZI 21250518 IC50 = 10600 nM T84631 CCY2M5 21366447 IC50 = 76 nM T84631 C27VLD 21366448 IC50 = 24 nM T84631 C1JQY7 21366475 IC50 = 15 nM T84631 C82SUW 21366478 IC50 = 8 nM T84631 CSG82H 21366479 IC50 = 7 nM T84631 CP0CR1 21366482 Ki = 0.7 nM T84631 CNTI15 21366511 IC50 = 143 nM T84631 C5S8ZW 21366513 IC50 = 24 nM T84631 CNC0E1 21366553 IC50 = 81 nM T84631 C9GAE1 21366554 IC50 = 39 nM T84631 C1CVM9 21366560 Ki = 5.2 nM T84631 C2LJ6Y 21366561 IC50 = 11 nM T84631 CQM6Y9 21366562 Ki = 4.1 nM T84631 C59WZX 21366563 IC50 = 10 nM T84631 C0H8KE 21366566 IC50 = 27 nM T84631 C67QCO 21366574 IC50 > 11000 nM T84631 CS2L1Y 21366575 IC50 = 483 nM T84631 CX1WM9 21366579 IC50 = 1650 nM T84631 C5XU1Y 21366636 Ki = 1.4 nM T84631 C0MXT9 21366640 Ki = 1.9 nM T84631 C0H3EX 21366644 Ki = 1 nM T84631 CYVC46 21366645 Ki = 1.2 nM T84631 C8OL1C 21366646 Ki = 1.8 nM T84631 C0U5PX 21366647 IC50 = 3 nM T84631 CP91WB 21366649 IC50 = 7 nM T84631 C8BLF5 21366650 IC50 = 4 nM T84631 CR8QB1 21366651 IC50 = 7 nM T84631 CKE17U 21366652 IC50 = 2 nM T84631 CV16OC 21366654 Ki = 0.9 nM T84631 CTND64 21578548 Ki = 27558 nM T84631 C7Z8YR 21845821 Ki = 6.31 nM T84631 C3HY2D 21845878 Ki = 1258.93 nM T84631 CI0SJ2 21967345 Ki = 5 nM T84631 CK5I4A 21968289 Ki = 170 nM T84631 CXV3I1 22017200 Ki = 320 nM T84631 C0MI4Y 22038750 Ki > 7500 nM T84631 CAS92P 22038873 Ki = 12200 nM T84631 CJ81IS 22039255 Ki = 730 nM T84631 C7VD8G 22039455 Ki = 790 nM T84631 CD2I7L 22039678 Ki = 1400 nM T84631 CK6E8W 22052309 Ki = 48 nM T84631 C4QDG0 22052319 Ki = 50 nM T84631 C0OE1R 22052320 Ki = 29 nM T84631 CX0FL5 22052323 Ki = 13 nM T84631 CHQ1R5 22052325 Ki = 61 nM T84631 CXPM37 22052326 Ki = 316 nM T84631 C6T8ZN 22052336 Ki = 86 nM T84631 C1YH0L 22052339 Ki = 54 nM T84631 COW3F2 22052347 Ki = 140 nM T84631 CSJW40 22052358 Ki = 25 nM T84631 CTNL12 22052361 Ki = 12.59 nM T84631 C4L1XD 22052368 Ki = 106 nM T84631 CC52AE 22052371 Ki = 39.81 nM T84631 C29PIU 22052373 Ki = 37 nM T84631 CA5T8Z 22052377 Ki = 1763 nM T84631 C8C7PW 22052392 Ki = 233 nM T84631 C9L5AD 22052419 Ki = 263 nM T84631 CC6Z8A 22052426 Ki = 19.95 nM T84631 CJ9W2M 22052436 Ki = 76 nM T84631 C8D7FS 22052452 Ki = 28 nM T84631 CTO8P4 22052453 Ki = 398.11 nM T84631 CV7O1I 22052465 Ki = 1554 nM T84631 C17HKB 22052478 Ki = 20 nM T84631 C1O9GL 22052482 Ki = 39.81 nM T84631 CGNH32 22052484 Ki = 75 nM T84631 CQ5VT0 22052485 Ki = 44 nM T84631 CN6YR8 22052493 Ki = 314 nM T84631 C7FYD1 22086911 Ki = 2.8 nM T84631 C5VIU4 22086968 Ki = 1.7 nM T84631 CYEU57 22086972 Ki = 0.53 nM T84631 C5K6SW 22086973 Ki = 0.55 nM T84631 CQC51W 22086974 Ki = 0.35 nM T84631 C9LI4W 22086975 Ki = 0.25 nM T84631 CB6IP5 22086976 Ki = 0.04 nM T84631 C3O8DP 22086978 Ki = 1.5 nM T84631 CDVH80 22086981 Ki = 0.35 nM T84631 CLH7A0 22086982 Ki = 0.15 nM T84631 C17KGP 22086987 Ki = 1.3 nM T84631 CG4ZH7 22086988 Ki = 0.31 nM T84631 CVM24X 22086990 Ki = 2.8 nM T84631 CJ5D8V 22086991 Ki = 1.4 nM T84631 C5V2HO 22086992 Ki = 1.9 nM T84631 CZ5O0I 22087006 Ki = 0.85 nM T84631 COK2S6 22087007 Ki = 0.81 nM T84631 CJ8D4K 22087014 Ki = 2.1 nM T84631 CKT23G 22125586 Ki = 30 nM T84631 CA3I4Y 22280766 Ki = 4.6 nM T84631 C40XEN 22313515 Ki = 450 nM T84631 CH9E3I 22313526 Ki = 560 nM T84631 C04OMK 22318549 Ki = 1 nM T84631 CS01PB 22318550 Ki = 23 nM T84631 CSQ96D 22336121 IC50 = 19.41 nM T84631 C7R9CD 22336127 IC50 = 0.64 nM T84631 C1R9CX 22336133 IC50 = 5.22 nM T84631 CHOQ30 22336142 IC50 = 8.15 nM T84631 CVG29W 22336143 IC50 = 0.12 nM T84631 CB7N4X 22336146 IC50 = 0.15 nM T84631 C8URK9 22336148 IC50 = 59 nM T84631 C3QEL8 22336150 IC50 = 0.15 nM T84631 C5O7VB 22336151 IC50 = 0.04 nM T84631 C19NAE 22336153 IC50 = 0.35 nM T84631 CHG0A5 22336163 IC50 = 1.65 nM T84631 CTOR48 22336172 IC50 = 0.45 nM T84631 C51FCG 22336174 IC50 = 0.23 nM T84631 CXZ92L 22336180 IC50 = 1.9 nM T84631 C85UYR 22336181 IC50 = 0.05 nM T84631 CU3T0V 22394327 Ki = 2900 nM T84631 CN6P9I 22394409 Ki = 18 nM T84631 CYLS84 22394472 Ki = 2997 nM T84631 CIT61O 22458350 IC50 = 3.6 nM T84631 CCD92W 22458360 IC50 = 3120 nM T84631 CRHI62 22458366 IC50 = 184 nM T84631 CCM12G 22458368 IC50 = 270 nM T84631 CT2IM0 22458374 IC50 = 920 nM T84631 CYOX21 22458381 IC50 = 880 nM T84631 COLY72 22556932 Ki = 2 nM T84631 C2V1NP 22556955 Ki = 2 nM T84631 C4YL7S 22556963 Ki = 0.7 nM T84631 C9VXC8 22556983 Ki = 20 nM T84631 CY4J8E 22596314 IC50 = 12 nM T84631 CLA45C 22596321 IC50 = 48 nM T84631 CF2RK6 22596324 IC50 = 2.5 nM T84631 C2KTB6 22596330 IC50 = 1.9 nM T84631 C9FVL3 22596339 IC50 = 49 nM T84631 C1B0NE 22596349 IC50 = 1.8 nM T84631 CC7LV3 22596380 IC50 = 4.4 nM T84631 CTG8D5 22596389 IC50 = 2.5 nM T84631 CZ4T5U 22596395 IC50 = 7.7 nM T84631 C32GEK 22596430 IC50 = 4.6 nM T84631 CA3FT7 22612508 Ki = 390 nM T84631 CUXK90 22628841 Ki = 60 nM T84631 C4W0GT 22713568 Ki > 10000 nM T84631 CJY09H 22861145 Ki = 130016.96 nM T84631 CN3ZI2 22883539 Ki = 90 nM T84631 CW8EH6 22883547 Ki = 39 nM T84631 CA3N9L 22883564 Ki = 31 nM T84631 C9DB7V 22883573 Ki = 120 nM T84631 CVZ15N 22883583 Ki = 88 nM T84631 C1R0UD 22883585 Ki = 26 nM T84631 C13-JAN 22883594 Ki = 3 nM T84631 C1KG8E 22945874 IC50 = 110 nM T84631 C3VZ7S 23283289 Ki = 19000 nM T84631 CV5NL8 23283331 Ki = 30000 nM T84631 C2K7VO 23396194 Ki = 588 nM T84631 CU01TZ 23396195 Ki = 241 nM T84631 CR6CQ9 23396199 Ki = 50 nM T84631 CY32CO 23396230 Ki = 37 nM T84631 CXD84O 23396232 Ki = 125 nM T84631 C9BUH2 23396254 Ki = 630.96 nM T84631 CEVA63 23396255 Ki = 36 nM T84631 C71ZYM 23396256 Ki = 71 nM T84631 CG3VZ4 23396258 Ki = 41 nM T84631 C3Z2EI 23396259 Ki = 4605 nM T84631 C5B8YE 23396265 Ki > 10000 nM T84631 C16WGD 23396266 Ki > 10000 nM T84631 CW3VI5 23396282 Ki = 1931 nM T84631 C3EH5R 23396283 Ki = 2494 nM T84631 C2P7KJ 23396286 Ki = 1552 nM T84631 C0Z3IW 23396287 Ki = 100 nM T84631 CI76UO 23396288 Ki = 124 nM T84631 CO63QT 23396289 Ki = 3162.28 nM T84631 C9ZAU2 23396290 Ki = 199.53 nM T84631 C0GWO4 23396291 Ki = 307 nM T84631 C7ICP0 23396292 Ki = 199.53 nM T84631 CCA13I 23396298 Ki = 39 nM T84631 C9VZK5 23396327 Ki = 4531 nM T84631 CN1H6K 23396328 Ki > 10000 nM T84631 CR2Y5O 23442128 Ki = 650 nM T84631 CQ70HF 23586156 IC50 = 995 nM T84631 C1JXS8 23634638 Ki = 1.7 nM T84631 C0W2EP 23634640 Ki = 0.33 nM T84631 CD7C1W 23634756 Ki = 9.6 nM T84631 C2KJ0P 23634757 Ki = 6.7 nM T84631 C6Z9WS 23634758 Ki = 2 nM T84631 C92VIM 23634877 Ki = 1.7 nM T84631 CY3NC8 23634878 Ki = 0.31 nM T84631 CP6Y7K 23634881 Ki = 0.63 nM T84631 C61GCE 23635132 Ki = 0.48 nM T84631 C75GTN 23635133 Ki = 0.85 nM T84631 C7HOG9 23635260 Ki = 1.1 nM T84631 CR9BK5 23635261 Ki = 1584.89 nM T84631 CDHQ47 23635262 Ki = 180 nM T84631 C1KCZ6 23635264 Ki = 0.5 nM T84631 CR8AK4 23635386 Ki = 2.1 nM T84631 C7U9XO 23635500 Ki = 0.54 nM T84631 C8URE5 23635503 Ki = 4.8 nM T84631 CH9F4R 23635626 Ki = 0.67 nM T84631 CA07TV 23635750 Ki = 0.25 nM T84631 CA7Q4T 23635752 Ki = 610 nM T84631 C06FJI 23635753 Ki = 6 nM T84631 CTS9W8 23636240 Ki = 0.25 nM T84631 C50TMW 23636367 Ki = 3.9 nM T84631 C04CKF 23636368 Ki = 7.6 nM T84631 CZO8U6 23636369 Ki = 0.08 nM T84631 C10EHQ 23636370 Ki = 0.3 nM T84631 C7JF0K 23636371 Ki = 0.07 nM T84631 CCD8R5 23644670 Ki = 82 nM T84631 CEL6C2 23644671 Ki = 0.38 nM T84631 C6KY5R 23644672 Ki = 0.66 nM T84631 CJ1QC3 23646071 Ki = 7 nM T84631 CXIY21 23646108 Ki = 346 nM T84631 C6F3VD 23646109 Ki = 56 nM T84631 C83WUS 23646110 Ki = 2720 nM T84631 C4SB7E 23646111 Ki = 22 nM T84631 C6WB0S 23646112 Ki = 136 nM T84631 CM29UX 23646113 Ki = 57 nM T84631 CN18XI 23646114 Ki = 73 nM T84631 CET26V 23646115 Ki = 27 nM T84631 C1V0EW 23646116 Ki = 24 nM T84631 C1NO3E 23646117 Ki = 4100 nM T84631 C0GT7A 23646118 Ki = 15 nM T84631 CZ7U0G 23646119 Ki = 11 nM T84631 CF52TJ 23646120 Ki = 39000 nM T84631 CE71BT 23646121 Ki = 3 nM T84631 CTD16K 23646122 Ki = 2 nM T84631 CZ8CT7 23646123 Ki < 1 nM T84631 C5FG7J 23646124 Ki = 1 nM T84631 C4SL3W 23646125 Ki = 1 nM T84631 CQA78Z 23646126 Ki < 1 nM T84631 C8VA1Z 23646127 Ki = 60 nM T84631 CQ21XZ 23646128 Ki = 72 nM T84631 C16JDI 23646129 Ki = 63 nM T84631 CUX4J8 23646130 Ki = 1 nM T84631 CN7X8I 23646131 Ki = 2 nM T84631 CNK52C 23646132 Ki = 10600 nM T84631 CE5QN2 23646133 Ki = 50 nM T84631 CT9U3L 23646134 Ki = 320 nM T84631 CW2GJ6 23646135 Ki = 2060 nM T84631 CC3YP4 23646136 Ki = 160 nM T84631 C38SAT 23646137 Ki = 40 nM T84631 CXD31S 23646138 Ki = 82 nM T84631 C92MUL 23646153 Ki = 1.6 nM T84631 CJ9OA4 23646154 Ki = 0.13 nM T84631 CP23GI 23646155 Ki = 0.11 nM T84631 CH1LX7 23646156 Ki < 0.1 nM T84631 C83QCW 23646157 Ki = 0.34 nM T84631 CX8FL0 23646158 Ki = 0.12 nM T84631 C05YBQ 23646159 Ki = 0.22 nM T84631 CYB83X 23646160 Ki = 0.64 nM T84631 CZS9J8 23646161 Ki = 0.71 nM T84631 C3N8QU 23646162 Ki = 0.24 nM T84631 C7OC4K 23646163 Ki = 0.16 nM T84631 CA8EP1 23646164 Ki = 0.27 nM T84631 CVF49W 23646165 Ki = 0.34 nM T84631 CM94VT 23646166 Ki = 8.4 nM T84631 CY3CP9 23646167 Ki = 45 nM T84631 CIR80B 23646168 Ki = 1.5 nM T84631 C9OS8M 23646169 Ki = 2.1 nM T84631 CLKM63 23646170 Ki = 1.8 nM T84631 C08QUL 23646171 Ki = 0.82 nM T84631 CS80IC 23646172 Ki = 2.7 nM T84631 CZ9TO3 23646173 Ki = 12 nM T84631 CGS86R 23646174 Ki = 20 nM T84631 CGE2M7 23646175 Ki = 2 nM T84631 CK0X2L 23646176 Ki = 88 nM T84631 CX3GB9 23646177 Ki = 54 nM T84631 C07LKX 23646178 Ki = 47 nM T84631 C0IVO1 23646179 Ki = 2.6 nM T84631 CLC9F3 23646180 Ki = 1.2 nM T84631 CGVJ65 23646181 Ki = 0.18 nM T84631 C7MC5Y 23646182 Ki = 0.74 nM T84631 CGFT69 23646183 Ki = 2 nM T84631 C7P4VU 23646184 Ki = 0.18 nM T84631 C6Q1CR 23646185 Ki = 0.18 nM T84631 CKB59A 23646186 Ki = 0.12 nM T84631 CA0LC6 23646187 Ki = 0.2 nM T84631 CM01LP 23646188 Ki = 0.09 nM T84631 CA3U0I 23646189 Ki = 0.02 nM T84631 CIR65F 23646190 Ki = 0.03 nM T84631 CDK0P2 23646191 Ki = 0.04 nM T84631 CJ4U2X 23646192 Ki = 0.02 nM T84631 CMYI38 23646193 Ki = 0.42 nM T84631 CZ1KO7 23646194 Ki = 0.25 nM T84631 CPF54M 23646195 Ki = 0.29 nM T84631 CP84AB 23646196 Ki = 0.27 nM T84631 C2WK4G 23646197 Ki = 0.12 nM T84631 CC1FV9 23646198 Ki = 0.08 nM T84631 CG82YE 23646199 Ki = 0.27 nM T84631 C5KWB9 23646200 Ki = 5.4 nM T84631 CY8SQ7 23646201 Ki = 0.05 nM T84631 CCMZ94 23646202 Ki = 0.58 nM T84631 C08AOH 23646204 Ki = 0.26 nM T84631 C82COD 23646205 Ki = 0.31 nM T84631 CS5AL3 23646206 Ki = 0.2 nM T84631 C0EO5K 23646207 Ki = 0.65 nM T84631 CN1Q7D 23646208 Ki = 0.63 nM T84631 CP24HW 23646209 Ki = 2.5 nM T84631 C6UM7B 23646210 Ki = 1.3 nM T84631 C7NKV6 23646211 Ki = 26 nM T84631 CGB18F 23646212 Ki = 3 nM T84631 C5J3OT 23646213 Ki = 2.2 nM T84631 C3JF1O 23646214 Ki = 2.8 nM T84631 C75SDV 23646215 Ki = 14 nM T84631 C8G0NU 23646216 Ki = 6.1 nM T84631 C84HGM 23646217 Ki = 28 nM T84631 CATE50 23646218 Ki = 4 nM T84631 CC52RE 23646219 Ki = 7 nM T84631 C7CZ2J 23646220 Ki = 18 nM T84631 CLDZ20 23646221 Ki = 19 nM T84631 CM7X3R 23646222 Ki = 5.6 nM T84631 CG3ZB2 23646223 Ki = 160 nM T84631 CQS7X6 23646224 Ki = 45 nM T84631 CHAD98 23646225 Ki = 36 nM T84631 C8XZ3J 23646226 Ki = 72 nM T84631 CP9A1B 23646227 Ki = 810 nM T84631 CJS63R 23646228 Ki = 2600 nM T84631 CJN96Y 23646229 Ki = 79 nM T84631 C01VKP 23646230 Ki = 1100 nM T84631 CL14AX 23646231 Ki = 120 nM T84631 C96UDO 23646233 Ki = 2.5 nM T84631 C6RM8B 23646234 Ki = 47 nM T84631 C2U0RB 23646236 Ki = 4 nM T84631 CPMW70 23646237 Ki = 740 nM T84631 CS5CV9 23646239 Ki = 71 nM T84631 CV1HY5 23646241 Ki = 22 nM T84631 C6BG3M 23646243 Ki = 280 nM T84631 CU2V7C 23646245 Ki = 2020 nM T84631 C93IYD 23646247 Ki = 5360 nM T84631 C5LQ0H 23646249 Ki = 450 nM T84631 CS68GZ 23646251 Ki > 8000 nM T84631 C7FEL6 23646252 Ki > 8000 nM T84631 C3ZAY1 23646254 Ki > 8000 nM T84631 C6EF4Y 23646256 Ki = 3240 nM T84631 CKM7Y4 23646258 Ki = 410 nM T84631 C0UMW5 23646268 Ki = 2700 nM T84631 C2RV5T 23646269 Ki = 5700 nM T84631 C4YPZ3 23646288 Ki = 2 nM T84631 CD7YW3 23646289 Ki = 0.27 nM T84631 C25LRJ 23646290 Ki = 0.25 nM T84631 CI0W3O 23646291 Ki = 0.34 nM T84631 CM5VS7 23646292 Ki = 0.2 nM T84631 CQI1G4 23646293 Ki = 0.3 nM T84631 CY96RK 23646294 Ki = 0.4 nM T84631 CRX19I 23646295 Ki = 0.1 nM T84631 CP4GN0 23646296 Ki = 0.2 nM T84631 CI04YH 23646297 Ki = 0.53 nM T84631 CB3JK7 23646298 Ki = 0.52 nM T84631 COV42F 23646299 Ki = 0.54 nM T84631 CJR4X5 23646300 Ki = 0.15 nM T84631 CN2D0X 23646301 Ki = 0.55 nM T84631 C8GX6A 23646302 Ki = 0.86 nM T84631 CUF86C 23646303 Ki = 1.14 nM T84631 CU1Z9L 23646304 Ki = 0.08 nM T84631 C69ZVT 23646306 Ki = 0.02 nM T84631 CZ6GK2 23646308 Ki = 0.05 nM T84631 C5NF0J 23646310 Ki = 0.5 nM T84631 C2XQ7C 23646311 Ki = 0.35 nM T84631 CCRD27 23646312 Ki = 0.17 nM T84631 CLC17N 23646313 Ki = 0.5 nM T84631 CS2RE4 23646314 Ki = 0.18 nM T84631 C1WE6B 23646315 Ki = 0.21 nM T84631 CM4NQ5 23646316 Ki = 0.35 nM T84631 CAN6D5 23646317 Ki = 0.11 nM T84631 CKO58P 23646318 Ki = 0.22 nM T84631 C25WIE 23646319 Ki = 3.2 nM T84631 CLB4D5 23646320 Ki = 0.77 nM T84631 CDYF29 23646329 IC50 = 85000 nM T84631 CQB29J 23646453 Ki = 5600 nM T84631 C74AMD 23646454 Ki = 13300 nM T84631 CZ7JM9 23646455 Ki = 2300 nM T84631 CD9UH7 23646456 Ki = 2600 nM T84631 CX5S3K 23646457 Ki = 9100 nM T84631 CEH94J 23646458 Ki = 15300 nM T84631 C1DRZ7 23646459 Ki = 1500 nM T84631 CK64IY 23646460 Ki = 2200 nM T84631 CSY57G 23646463 Ki > 74000 nM T84631 CZ48JL 23646472 Ki = 10000 nM T84631 CJR27Q 23646473 Ki = 10000 nM T84631 CY5SE6 23646474 Ki = 156 nM T84631 C73ZDQ 23646475 Ki = 1053 nM T84631 C7CXM5 23646476 Ki = 285 nM T84631 C54VIZ 23646526 Ki = 110 nM T84631 CSL27U 23646528 Ki = 4830 nM T84631 CJ5CZ8 23646530 Ki = 14480 nM T84631 C7SZ4N 23646532 Ki = 180 nM T84631 CM74YK 23646533 Ki = 1310 nM T84631 CB1GR0 23646534 Ki = 3520 nM T84631 CSFH79 23646622 Ki = 440 nM T84631 C35HJA 23646623 Ki = 520 nM T84631 C7E4SA 23646732 Ki = 130 nM T84631 C4Z6FV 23647193 Ki = 103 nM T84631 C1L9VZ 23647194 Ki = 48 nM T84631 CU2Z6T 23647195 Ki = 225 nM T84631 CSG4O2 23647196 Ki = 345 nM T84631 CWHX79 23647197 Ki = 839 nM T84631 CC29KT 23647198 Ki = 12 nM T84631 CWCR31 23647199 Ki = 2730 nM T84631 CA52KT 23647200 Ki = 287 nM T84631 C9AG8L 23647650 Ki = 0.008 nM T84631 CI6N8M 23647676 Ki > 5000 nM T84631 C2QNL5 23647679 Ki = 3.4 nM T84631 CEP2K3 23647680 Ki = 1.5 nM T84631 CS08RA 23647681 Ki = 20 nM T84631 CQDG25 23647682 Ki = 5.7 nM T84631 CJC10T 23648140 Ki = 3 nM T84631 CC1Z9L 23648141 Ki = 5.7 nM T84631 C5ZP9A 23648142 Ki = 4.9 nM T84631 CR1BX3 23648143 Ki = 2.4 nM T84631 CARL42 23648144 Ki = 1.7 nM T84631 COI95T 23648145 Ki = 92 nM T84631 CM20FT 23648146 Ki = 14 nM T84631 CY75HR 23648147 Ki = 0.61 nM T84631 C2XIJ7 23648148 Ki = 0.73 nM T84631 C8F4ET 23648149 Ki = 0.67 nM T84631 C9HKT7 23648150 Ki = 0.7 nM T84631 CQ0RX9 23648151 Ki = 0.41 nM T84631 CM16WB 23648152 Ki = 0.26 nM T84631 C8PO4L 23648153 Ki = 0.57 nM T84631 CV6LR5 23648154 Ki = 0.87 nM T84631 CJ24TP 23648155 Ki = 0.26 nM T84631 CRW32H 23648156 Ki = 3.9 nM T84631 CH1D5R 23648157 Ki = 8.8 nM T84631 CU78RG 23648158 Ki = 29 nM T84631 C81PHJ 23648159 Ki = 6.6 nM T84631 CG3W5Q 23661706 IC50 > 30000 nM T84631 C9O1MH 23704948 IC50 > 5000 nM T84631 CKH4O5 24180463 Ki = 0.5 nM T84631 C7AYO1 24748789 IC50 = 20000 nM T84631 CVO5L6 24748791 IC50 = 13700 nM T84631 CUAY58 24749175 IC50 = 100000 nM T84631 C69OVW 24752832 IC50 = 16 nM T84631 CI93ZB 24752833 IC50 = 13 nM T84631 C3S1MT 24773377 Ki = 1.4 nM T84631 CF5I9O 24773378 Ki = 2255 nM T84631 CW8MT6 24773379 Ki = 4.1 nM T84631 CEQA82 24773380 Ki = 690 nM T84631 C93BFM 24773469 Ki = 4.9 nM T84631 C6N2IV 24773892 Ki = 8.1 nM T84631 CQTD47 24773893 Ki = 147 nM T84631 C6H7KF 24773969 Ki = 4.4 nM T84631 CGB15F 24773970 Ki = 231 nM T84631 C4CN1H 24774292 Ki > 14400 nM T84631 CO5JE3 24774293 Ki = 6850 nM T84631 CD6HV2 24774371 Ki = 26 nM T84631 CWX96Z 24774372 Ki = 22.9 nM T84631 CO2U9L 24774373 Ki = 6.4 nM T84631 CSW54F 24794406 Ki = 5.5 nM T84631 C8X5FS 24836819 Ki = 0.021 nM T84631 CJSO87 24849206 Ki = 7 nM T84631 CF7VA8 24858772 Ki = 1050 nM T84631 C6W5XL 24858773 Ki = 9270 nM T84631 CES0Y3 24858774 Ki = 15900 nM T84631 C9N8CR 24858929 Ki = 1940 nM T84631 C7QK4H 24858930 Ki = 5710 nM T84631 CWX43I 24858931 Ki = 58700 nM T84631 CNAG78 24858932 Ki = 139000 nM T84631 C8RHA3 24858933 Ki = 33200 nM T84631 C0UA9T 24860449 IC50 > 50000 nM T84631 C52CJA 24860451 IC50 > 50000 nM T84631 COX4A7 24873356 Ki = 4500 nM T84631 CYU34A 24881188 IC50 = 910 nM T84631 C9R2QI 24881190 IC50 = 460 nM T84631 C70AFO 24881191 IC50 = 54 nM T84631 C3KRV6 24881192 IC50 = 6.9 nM T84631 CO06JI 24881193 IC50 = 170 nM T84631 C2ON8C 24881194 IC50 = 56 nM T84631 CB20OY 24881251 IC50 = 160 nM T84631 C0FY1U 24881252 IC50 = 1400 nM T84631 CU6NH0 24881253 IC50 = 56 nM T84631 C87LAW 24881255 IC50 = 37 nM T84631 CDH1E3 24881256 IC50 = 300 nM T84631 C9PHM0 24882178 IC50 = 12 nM T84631 CY61BZ 24882254 IC50 = 23 nM T84631 C2RA7O 24882255 IC50 = 120 nM T84631 CE2U6A 24882256 IC50 = 31 nM T84631 C62GNZ 24882257 IC50 = 230 nM T84631 CT26DH 24882258 IC50 = 170 nM T84631 CKWT73 24882259 IC50 = 1600 nM T84631 CKJ7M2 24882363 IC50 = 50 nM T84631 CYJI62 24936113 Ki < 0.1 nM T84631 CYRU05 24936173 IC50 = 1.7 nM T84631 CQ52VL 24936196 Ki < 0.4 nM T84631 CY7BX0 24936197 Ki < 0.3 nM T84631 C7H5DI 24936198 Ki = 0.2 nM T84631 C3BD4T 24997732 Ki = 55 nM T84631 CN0ZW3 24999867 Ki > 1000 nM T84631 CEM32W 25001205 Ki > 1000 nM T84631 CJ84TQ 25015739 IC50 = 8.6 nM T84631 CAO2V4 25030840 Ki = 19000 nM T84631 CU82IO 25030929 Ki = 11200 nM T84631 C7MCT6 25031099 Ki = 2100 nM T84631 C5PO7A 25031100 Ki = 18000 nM T84631 CH7Z1K 25031101 Ki = 8200 nM T84631 CEW9X2 25031102 Ki = 6100 nM T84631 C9NC4S 25031541 Ki = 10000 nM T84631 CK5R8Q 25032200 Ki = 2500 nM T84631 CG8HY2 25032202 Ki = 15000 nM T84631 CH76XK 25032204 Ki = 26000 nM T84631 CN23DH 25049955 IC50 = 0.8 nM T84631 CZ78XH 25049956 IC50 = 0.54 nM T84631 CVS5A8 25049959 IC50 = 0.48 nM T84631 CO4PK0 25050108 IC50 = 0.38 nM T84631 CJR65Q 25050945 IC50 = 6.1 nM T84631 C29CKQ 25050946 IC50 = 2.1 nM T84631 CY61SV 25051116 IC50 = 5.6 nM T84631 CX5P3Q 25051117 IC50 = 3.5 nM T84631 CQK9R2 25051277 IC50 = 2.9 nM T84631 CYG9R7 25051278 IC50 = 2 nM T84631 CP0GX3 25051281 IC50 = 0.93 nM T84631 CO1Q3B 25051600 IC50 = 4.1 nM T84631 CR81PB 25052256 IC50 = 1.3 nM T84631 CBG9P4 25052257 IC50 = 2.3 nM T84631 C4PGS3 25052258 IC50 = 10 nM T84631 C16GLV 25052749 IC50 = 10 nM T84631 C07BZQ 25107507 Ki = 50300 nM T84631 CK3FM6 25107508 Ki = 31600 nM T84631 CN3I9J 25107569 Ki = 112000 nM T84631 CB6H7T 25107570 Ki = 2670 nM T84631 CC40FO 25107571 Ki = 112000 nM T84631 C1QC4Y 25107572 Ki = 16000 nM T84631 CKJ04T 25107573 Ki = 27700 nM T84631 CN8Y0B 25107634 Ki = 9590 nM T84631 C84XCZ 25107635 Ki = 16600 nM T84631 CCY26A 25107636 Ki = 29700 nM T84631 CO03GM 25107637 Ki = 29500 nM T84631 CNR43C 25107638 Ki = 12100 nM T84631 CDAC04 25107705 Ki = 33800 nM T84631 CYS45L 25107706 Ki = 43100 nM T84631 CYS98D 25107707 Ki = 49600 nM T84631 CRV78W 25107708 Ki = 11900 nM T84631 CF85WU 25107709 Ki = 18000 nM T84631 C23YAU 25107770 Ki = 11800 nM T84631 CQZ70E 25107771 Ki = 35400 nM T84631 CEK7G5 25107772 Ki = 74700 nM T84631 C3V7JU 25107773 Ki = 31700 nM T84631 C4LUT7 25113610 Ki = 9 nM T84631 CPBC45 25138134 IC50 = 110 nM T84631 CK2WL4 25138136 IC50 = 114 nM T84631 C1XY0D 25138137 IC50 = 430 nM T84631 C72JBP 25138138 IC50 = 650 nM T84631 CN10CG 25138139 IC50 = 13700 nM T84631 CB3FJ8 25138140 IC50 = 8.9 nM T84631 C9H0OL 25138141 IC50 = 118 nM T84631 CI8HE3 25138142 IC50 = 2.4 nM T84631 CW8B3G 25138143 IC50 = 9 nM T84631 CTE97L 25138144 IC50 = 290 nM T84631 CBV14T 25138145 IC50 = 17000 nM T84631 C2H4PJ 25166809 Ki = 5200 nM T84631 CG76TR 25181493 Ki = 360 nM T84631 CAX4Q1 25198342 Ki = 550 nM T84631 C16ILQ 25198493 Ki = 911 nM T84631 C6V9TD 25198622 Ki = 9800 nM T84631 CV46JB 25198623 Ki = 56 nM T84631 C4S0ZM 25210468 IC50 = 0.1 nM T84631 C5RJ1T 25210469 IC50 = 0.08 nM T84631 CV4O1F 25222767 Ki = 1450 nM T84631 C1W3CU 25222769 Ki = 9470 nM T84631 C1U9AE 25222771 Ki = 57 nM T84631 C15CWG 25222774 Ki = 260000 nM T84631 CH92VC 25222868 Ki = 2000 nM T84631 CEC04N 25222874 Ki = 2500 nM T84631 C8WG3X 25222971 Ki = 57000 nM T84631 CBP53A 25222975 Ki = 1000 nM T84631 CHTV50 25222977 Ki = 3870 nM T84631 CJ67WP 25222979 Ki = 767 nM T84631 C9WQU4 25222981 Ki = 512 nM T84631 CMY62V 25223085 Ki = 130 nM T84631 C4DK1F 25223087 Ki = 666 nM T84631 CL1WP8 25223089 Ki = 33800 nM T84631 CQ5OP1 25224184 Ki = 126000 nM T84631 CK5RQ4 25224186 Ki = 5200 nM T84631 CYD28U 25224296 Ki = 177 nM T84631 CFRU38 25224298 Ki = 548 nM T84631 CHD01M 25224300 Ki = 1270 nM T84631 C43UCD 25268815 IC50 = 9 nM T84631 CKM7Y8 25269170 Ki = 1.1 nM T84631 C37QUZ 25269526 IC50 = 3.2 nM T84631 CT0J3X 25270897 IC50 = 11.6 nM T84631 CU5YR1 41583852 IC50 > 200000 nM T84631 C62HGQ 42628060 Ki = 8 nM T84631 CJX5A6 42628061 Ki = 95 nM T84631 C3M0RO 42628062 Ki = 93 nM T84631 C19WJB 42628063 Ki = 31 nM T84631 CVAI06 42643068 Ki = 442 nM T84631 CUF74S 42643069 Ki = 162 nM T84631 CZ03OW 42643070 Ki = 112 nM T84631 CZ7M8C 42643120 Ki = 99 nM T84631 C0KN2D 42643121 Ki = 32 nM T84631 CL6GN4 42643122 Ki = 18 nM T84631 C6U1KC 42643173 Ki = 74 nM T84631 CC0XK4 42643174 Ki = 6 nM T84631 CV4EW7 42643175 Ki = 175 nM T84631 CN70MF 42643176 Ki = 1272 nM T84631 CHBR63 42643177 Ki = 11 nM T84631 CR1DQ2 42643222 Ki = 20 nM T84631 CH3IF2 42643277 Ki = 27 nM T84631 CRLZ98 42643388 Ki = 94 nM T84631 CQLA03 42643389 Ki = 132 nM T84631 C8ZJ0B 44156919 IC50 = 3280 nM T84631 CPX15D 44188281 IC50 = 7.1 nM T84631 CR8W6M 44200855 IC50 = 1.8 nM T84631 C4TZ2X 44201094 IC50 = 1.1 nM T84631 C9OMR4 44264598 Ki = 8700 nM T84631 CPRE58 44264710 Ki = 193 nM T84631 CA8N9H 44264719 Ki = 120 nM T84631 CW1G8N 44264814 Ki = 200 nM T84631 CF49JR 44264817 Ki = 59000 nM T84631 C6IDX1 44264832 Ki = 5000 nM T84631 CT40BD 44264834 Ki = 100000 nM T84631 C2XLN7 44264885 Ki = 7.1 nM T84631 CW4R8J 44264888 Ki = 2.2 nM T84631 CT2V6S 44264889 Ki = 3 nM T84631 CDNH87 44264912 Ki = 130 nM T84631 CZDW40 44264920 Ki = 3.3 nM T84631 C9RZ0O 44264921 Ki = 3.7 nM T84631 CXQ1H9 44264935 Ki = 14 nM T84631 C6O5VF 44264936 Ki = 2.5 nM T84631 CVBG38 44264940 Ki = 1.7 nM T84631 C63WPN 44264954 Ki = 34 nM T84631 CB3AQ1 44264955 Ki = 10 nM T84631 CGCI69 44264981 Ki = 1.2 nM T84631 C78WPK 44264995 Ki = 69 nM T84631 C01WIT 44265005 Ki = 15 nM T84631 C1BP7E 44265006 Ki = 11 nM T84631 CQNX29 44265034 Ki = 5.5 nM T84631 CQGC19 44265371 Ki = 43 nM T84631 CW6G5E 44271568 Ki = 2 nM T84631 CD2Z4T 44271573 Ki = 2 nM T84631 C65YHR 44271609 Ki = 25 nM T84631 CA18XV 44271621 Ki = 180 nM T84631 C13CDQ 44271631 Ki = 2 nM T84631 CA53QR 44271633 Ki = 35 nM T84631 C8BRO7 44271634 Ki = 48 nM T84631 C0SNH2 44271651 Ki = 75 nM T84631 CM4HK1 44271680 Ki = 1 nM T84631 C8U9EQ 44271692 Ki = 80 nM T84631 CC8G0D 44271702 Ki = 75 nM T84631 C4A5XW 44271749 Ki = 14 nM T84631 C9TD2K 44271760 Ki = 135 nM T84631 CU51BQ 44271777 Ki = 9 nM T84631 C7AS8L 44271778 Ki = 10 nM T84631 CMCS75 44272530 Ki = 36 nM T84631 C6GRO0 44272532 Ki = 5.8 nM T84631 C96TGO 44272560 Ki = 600 nM T84631 C65SNR 44272562 Ki = 3.1 nM T84631 C8CJI6 44272581 Ki = 150 nM T84631 CKZ6O0 44272690 Ki > 338 nM T84631 CB64EA 44272825 Ki = 1810 nM T84631 C1B9MI 44273291 IC50 = 70 nM T84631 C05TZL 44273376 IC50 = 66 nM T84631 C86OEF 44273389 IC50 = 22 nM T84631 CWU7G4 44273492 IC50 = 114 nM T84631 C1Z2QU 44273493 Ki = 2.5 nM T84631 C6ABM8 44273514 IC50 = 23 nM T84631 CW59QS 44273576 IC50 = 36 nM T84631 C8H0FK 44273592 IC50 = 92 nM T84631 CP32GC 44273614 IC50 = 430 nM T84631 CH3S8F 44273615 IC50 = 40 nM T84631 CYUQ93 44273643 IC50 = 13 nM T84631 C7EK0N 44273644 IC50 = 15 nM T84631 CV9C7T 44273645 Ki = 2.9 nM T84631 CR5A3C 44273666 IC50 = 108 nM T84631 CE3C6Q 44273679 IC50 = 26 nM T84631 CKUI85 44273680 IC50 = 380 nM T84631 C2S5UM 44273701 Ki = 1.1 nM T84631 CI9QM8 44273702 Ki = 0.5 nM T84631 CQ0HZ4 44273703 Ki = 0.3 nM T84631 CRA47X 44273704 IC50 = 39 nM T84631 CR6U4L 44273709 IC50 = 75 nM T84631 CZC9Q2 44273733 IC50 = 130 nM T84631 CJP8C0 44273734 IC50 = 112 nM T84631 CC30SE 44273735 IC50 = 215 nM T84631 CV13XP 44273736 IC50 = 94 nM T84631 CIQP84 44273737 IC50 = 131 nM T84631 C1HC0I 44273738 IC50 = 88 nM T84631 CZ5T6O 44273748 IC50 = 2100 nM T84631 C0A4ME 44273753 IC50 = 166 nM T84631 C2DJG4 44273754 Ki = 1.8 nM T84631 C8C1WF 44273817 IC50 = 3600 nM T84631 CCJN68 44273818 IC50 = 54000 nM T84631 CUG08B 44273828 IC50 = 680 nM T84631 CR3V4S 44273853 IC50 = 5200 nM T84631 CN4HE5 44273854 IC50 = 2900 nM T84631 C90AKQ 44273901 IC50 = 1100 nM T84631 CM3F7J 44273935 Ki = 1.1 nM T84631 CY4V8B 44273945 Ki = 2.8 nM T84631 C8ON3U 44273946 IC50 = 80 nM T84631 CI93OZ 44273947 IC50 = 48 nM T84631 CMD47X 44274011 Ki = 3.2 nM T84631 CL7NY5 44274017 Ki = 1.5 nM T84631 C68AOF 44274019 IC50 = 27 nM T84631 C7D5GB 44274020 IC50 = 47 nM T84631 C20PYG 44274030 IC50 = 110 nM T84631 C2BF3P 44274045 IC50 = 58 nM T84631 C41EMW 44274046 Ki = 0.5 nM T84631 CBAD49 44274051 IC50 = 479 nM T84631 CA10KD 44274052 IC50 = 377 nM T84631 C89BIR 44274053 IC50 = 34 nM T84631 CP1GC0 44274058 Ki = 1.8 nM T84631 C7I2DQ 44274065 IC50 = 7800 nM T84631 CI9E6O 44274072 IC50 = 13 nM T84631 COHA75 44274088 IC50 = 41 nM T84631 CMG90C 44274089 IC50 = 2 nM T84631 C6GKD2 44274282 IC50 = 22 nM T84631 CO7Z3E 44274843 Ki = 0.3 nM T84631 C7FP2X 44274865 Ki = 0.28 nM T84631 CNZ83L 44274886 Ki = 4 nM T84631 C9UP2G 44274929 Ki = 0.1 nM T84631 C9WDV8 44274930 Ki = 0.31 nM T84631 C3U8OC 44274931 Ki = 0.4 nM T84631 C2U5SO 44274945 Ki = 58 nM T84631 C5VE6G 44275194 Ki = 0.2 nM T84631 CT2J0P 44275195 Ki = 5 nM T84631 C42RVS 44275227 Ki = 13 nM T84631 CQ12EP 44275238 Ki = 74 nM T84631 C3OM8S 44275239 Ki = 0.1 nM T84631 CGOH67 44275240 Ki = 1.3 nM T84631 CU52WR 44275243 Ki = 8 nM T84631 C2HO4D 44275249 Ki = 0.028 nM T84631 C1N5GM 44275254 Ki = 0.46 nM T84631 CX1C4Q 44275257 Ki = 0.08 nM T84631 C9EKZ2 44275271 Ki = 64 nM T84631 C4TBU7 44275275 Ki = 50 nM T84631 C2D9YK 44275287 Ki = 2.2 nM T84631 CPBU68 44275289 Ki = 180 nM T84631 CL4D3K 44275297 Ki = 260 nM T84631 C3LS5P 44275326 Ki = 670 nM T84631 CHJC81 44275330 Ki = 34 nM T84631 C4SO5M 44275345 Ki = 150 nM T84631 CBA9T0 44275361 Ki = 17 nM T84631 CEWU09 44275365 Ki = 50 nM T84631 CVU1T9 44277085 IC50 > 2500 nM T84631 C19OGX 44278104 Ki = 385 nM T84631 C4A1ZJ 44282153 Ki > 10000 nM T84631 C5DZ4L 44282601 Ki > 10000 nM T84631 CRT93X 44282678 Ki > 10000 nM T84631 CA6X2L 44283195 Ki > 10000 nM T84631 CK29QN 44284451 IC50 = 7 nM T84631 CR09BC 44284461 IC50 = 362 nM T84631 CI65CK 44284478 IC50 = 35 nM T84631 CFJ9X2 44284522 IC50 = 245 nM T84631 CMU9A4 44284541 IC50 = 0.5 nM T84631 CI9H5W 44284543 IC50 = 5 nM T84631 CXK3M6 44284559 IC50 = 0.2 nM T84631 C6MUA4 44284604 IC50 = 759 nM T84631 C2JXL4 44284641 IC50 = 99 nM T84631 C96SRI 44284734 IC50 = 7 nM T84631 C36PXQ 44284752 IC50 = 99 nM T84631 CDAO90 44284753 IC50 = 664 nM T84631 C26YIW 44284754 IC50 = 628 nM T84631 C9DE2B 44284786 Ki = 0.18 nM T84631 CM4B7C 44284787 IC50 = 1.5 nM T84631 C41JHD 44284797 IC50 = 0.75 nM T84631 CUC1P9 44284803 IC50 = 2.6 nM T84631 CDM4W1 44284804 IC50 = 3 nM T84631 CEG25W 44284810 IC50 = 234 nM T84631 C4XE0Z 44284859 IC50 = 3.7 nM T84631 C2RCE1 44284893 IC50 = 9 nM T84631 C1IQY7 44284894 IC50 = 53 nM T84631 CR26VN 44284895 IC50 = 48 nM T84631 C31KIT 44284934 IC50 = 15 nM T84631 CU57SJ 44284940 IC50 = 17 nM T84631 C6Y7AO 44284957 IC50 = 18 nM T84631 C0KF4D 44284959 IC50 = 6470 nM T84631 CMZ71H 44284992 Ki = 0.58 nM T84631 CQ3N4P 44285111 IC50 = 13 nM T84631 C5NU9L 44285118 Ki = 13 nM T84631 CZ89KE 44285126 IC50 = 191 nM T84631 CFDP09 44285127 IC50 = 10 nM T84631 C9UP4E 44285152 IC50 = 4 nM T84631 CB45NT 44285154 IC50 = 215 nM T84631 CU9G2F 44285211 Ki = 2.6 nM T84631 C0FPN1 44285253 Ki = 7.2 nM T84631 C9N1ZL 44285281 Ki = 1.2 nM T84631 C5PX3O 44285312 Ki = 4.3 nM T84631 C9LRW8 44285352 Ki = 23 nM T84631 CQ82ZW 44286426 IC50 = 2500 nM T84631 COPR02 44286428 IC50 = 905 nM T84631 CS5U7F 44286453 IC50 = 447 nM T84631 CPK5M6 44286709 Ki = 69000 nM T84631 CQ2A3R 44286878 Ki = 66000 nM T84631 CJP7K9 44286879 Ki > 75000 nM T84631 CRK53N 44286978 Ki = 53000 nM T84631 C0DG5R 44287043 Ki = 92000 nM T84631 C63JTG 44287260 IC50 = 11000 nM T84631 CB9D2R 44287527 IC50 = 3000 nM T84631 CCXM09 44287610 IC50 = 550 nM T84631 CB8IQ5 44287628 IC50 = 27 nM T84631 CT4N0L 44287629 IC50 = 28 nM T84631 CS5D4G 44287745 IC50 = 15 nM T84631 CL5I1S 44287757 IC50 = 140 nM T84631 C3QD4W 44287797 Ki = 120000 nM T84631 C5W7SA 44287798 Ki = 29000 nM T84631 CX47AK 44287838 IC50 = 60000 nM T84631 C5Q9OJ 44287854 IC50 = 46 nM T84631 C5UT7J 44287855 IC50 = 20 nM T84631 C02ARM 44287937 Ki > 200000 nM T84631 CP90NM 44288029 Ki = 110000 nM T84631 CZRH12 44290033 IC50 = 21 nM T84631 CUY95P 44290108 IC50 = 7820 nM T84631 CS76AC 44290361 IC50 = 9900 nM T84631 C3WR2N 44290375 IC50 = 3.6 nM T84631 CMY82L 44290376 IC50 > 20000 nM T84631 CHL9Y6 44290377 IC50 > 100000 nM T84631 CLDH85 44290378 IC50 = 3600 nM T84631 CXO05N 44290379 IC50 > 200000 nM T84631 CCH40M 44290403 IC50 = 25 nM T84631 CJ20SI 44290431 IC50 = 22 nM T84631 C0E3FW 44290444 IC50 = 226 nM T84631 C9D7QK 44290445 IC50 = 623 nM T84631 CD8E0V 44290452 IC50 = 3.4 nM T84631 C9ZYO2 44290453 IC50 = 5.6 nM T84631 CUH6W4 44290457 IC50 = 16 nM T84631 CNWI90 44290501 IC50 > 200000 nM T84631 CBE24K 44290502 IC50 > 100000 nM T84631 C94BSK 44290516 IC50 = 20000 nM T84631 CAXB95 44290518 IC50 > 50000 nM T84631 C49EPA 44290519 IC50 = 2200 nM T84631 C37IJH 44290520 IC50 = 3700 nM T84631 CU17NH 44290529 IC50 = 5600 nM T84631 CC8YQ3 44290530 IC50 = 74 nM T84631 CN04WY 44290542 IC50 = 14000 nM T84631 CF8JK0 44290543 Ki = 11 nM T84631 C05EYJ 44290555 IC50 = 120 nM T84631 C10ANS 44290556 IC50 = 26000 nM T84631 CO9JQ0 44290557 Ki = 6 nM T84631 CY60EW 44290560 Ki = 2 nM T84631 C70XKC 44290569 Ki = 2.7 nM T84631 C9QS3I 44290584 Ki = 46 nM T84631 CUW14A 44290648 Ki = 4 nM T84631 COB93L 44290673 Ki = 69 nM T84631 C2UV6T 44290696 Ki = 8 nM T84631 C8LY1J 44290712 Ki = 20 nM T84631 C0SYK2 44290731 Ki = 0.4 nM T84631 CN6KP1 44290929 Ki > 1200 nM T84631 C0E1RV 44290930 Ki = 1 nM T84631 C8APX2 44290947 Ki = 0.5 nM T84631 CZ7PT1 44290965 Ki = 2 nM T84631 CTA7I1 44291034 Ki = 8 nM T84631 CH59WK 44291046 Ki = 0.89 nM T84631 CYFC04 44291049 Ki = 0.8 nM T84631 C7TNE0 44291050 Ki = 0.58 nM T84631 CC4RN5 44291077 Ki = 3 nM T84631 C0BKW7 44293012 Ki = 340 nM T84631 C18BMD 44293013 Ki = 620 nM T84631 CMN52F 44293014 Ki = 160 nM T84631 CQ0MU6 44293035 Ki = 620 nM T84631 C2RZ0Q 44293068 Ki = 97 nM T84631 C8ANR4 44293069 Ki > 1200 nM T84631 C4QNY6 44293089 Ki = 170 nM T84631 CWTU04 44293097 Ki > 1200 nM T84631 CID0Q1 44293197 Ki > 1200 nM T84631 CQ5M9L 44293198 Ki = 430 nM T84631 C4JI1E 44293369 Ki > 1200 nM T84631 C07IRQ 44293370 Ki > 1200 nM T84631 CX15SW 44293371 Ki > 1200 nM T84631 CK5H8X 44293458 Ki > 1200 nM T84631 CWV12E 44293459 Ki > 1200 nM T84631 CT7Q9E 44293503 Ki = 140 nM T84631 C2FMV6 44293504 Ki = 59 nM T84631 CV3NJ0 44293505 Ki = 250 nM T84631 C5IX3B 44293517 Ki > 1200 nM T84631 C9BT7Y 44293520 Ki = 140 nM T84631 CMG6H7 44293524 Ki = 270 nM T84631 C18JSA 44293525 Ki > 1200 nM T84631 CXV2U0 44293745 Ki = 120 nM T84631 CYHM09 44293746 Ki = 51 nM T84631 CKX76L 44294121 Ki = 1100 nM T84631 CWZ6Y0 44294144 Ki = 190 nM T84631 C5AZX1 44294161 Ki = 180 nM T84631 CQH6J3 44294201 Ki = 300 nM T84631 C5P8QF 44294202 Ki = 130 nM T84631 CI8V6A 44295540 Ki > 30000 nM T84631 CBD7K8 44295640 Ki = 2300 nM T84631 C39DAX 44295655 Ki = 2300 nM T84631 CJIA32 44295656 Ki > 30000 nM T84631 CJ9P3I 44295714 Ki = 17000 nM T84631 CPH39G 44295719 Ki = 24000 nM T84631 C46QHZ 44295721 Ki > 30000 nM T84631 C0O2PG 44295723 Ki = 10 nM T84631 CVYK28 44295735 Ki > 3000 nM T84631 CH0E5L 44295746 Ki > 30000 nM T84631 C0CDH2 44295750 Ki > 30000 nM T84631 C7F8HQ 44295757 Ki > 3000 nM T84631 C8G9EL 44295762 Ki = 26000 nM T84631 C2F7KZ 44295778 Ki > 30000 nM T84631 CH9TZ2 44295784 Ki = 490 nM T84631 C6U9CB 44295788 Ki = 1000 nM T84631 C7SN2O 44295812 Ki = 45 nM T84631 C1JYX7 44295834 Ki > 30000 nM T84631 CO4CV7 44295859 Ki = 1000 nM T84631 CQGD83 44295860 Ki = 4500 nM T84631 CSU4I8 44295861 Ki = 5900 nM T84631 CG17NR 44295877 Ki = 1800 nM T84631 C5S9RT 44295886 Ki = 2100 nM T84631 C0VBP5 44295901 Ki = 1700 nM T84631 CJCG97 44295904 Ki = 4600 nM T84631 CYFO56 44295908 Ki = 1700 nM T84631 C0N7OK 44295909 Ki = 1300 nM T84631 C4TQP8 44295912 Ki = 1700 nM T84631 CRZ24O 44295918 Ki = 17000 nM T84631 CMY02C 44295921 Ki = 1600 nM T84631 C2FK9M 44295923 Ki = 1100 nM T84631 CNI38U 44295960 Ki = 13200 nM T84631 C7JPH8 44295961 Ki = 2700 nM T84631 CN6UB9 44295962 Ki = 2500 nM T84631 C79ELR 44295964 Ki = 2400 nM T84631 CSW5Q1 44295971 Ki = 7500 nM T84631 CGDS36 44295996 Ki = 7800 nM T84631 C3ZL5P 44296008 Ki = 700 nM T84631 C1O3YJ 44296027 Ki = 20000 nM T84631 C8AY9O 44296035 Ki = 7600 nM T84631 CLK7N1 44296052 Ki = 8400 nM T84631 CQ51FN 44296074 Ki = 1200 nM T84631 CETN87 44296078 Ki = 300000 nM T84631 C3DG0L 44296128 Ki = 4 nM T84631 CPF86Z 44296129 Ki = 350 nM T84631 C38SDX 44296130 Ki = 4300 nM T84631 C1WU8B 44296135 Ki = 20 nM T84631 C3O6LY 44296148 Ki = 4100 nM T84631 CHI4G1 44296149 Ki = 10000 nM T84631 C6WNO3 44296150 Ki = 11000 nM T84631 C8WKO5 44296170 Ki = 15000 nM T84631 CV31AF 44296181 Ki > 5000 nM T84631 CW8N6G 44296281 Ki = 1900 nM T84631 CXL8T3 44296383 Ki = 3 nM T84631 C9AGW7 44297775 Ki = 290 nM T84631 C5HX1A 44297783 Ki = 2800 nM T84631 C4LMD2 44298298 Ki > 5000 nM T84631 CGBX35 44298541 Ki > 5000 nM T84631 C5YZ0H 44298559 Ki > 5000 nM T84631 CJE93G 44298563 Ki > 5000 nM T84631 CWA7D2 44298564 Ki > 5000 nM T84631 CYQN71 44298587 Ki > 5000 nM T84631 CCRS93 44298594 Ki > 5000 nM T84631 CW5NL8 44298595 Ki > 5000 nM T84631 C5ZIQ1 44298940 Ki > 5000 nM T84631 CSKI34 44298941 Ki > 5000 nM T84631 CB5UA1 44298971 Ki > 5000 nM T84631 CU3NP5 44298972 Ki > 5000 nM T84631 CERA27 44299040 Ki > 5000 nM T84631 C29MVU 44303719 Ki > 470000 nM T84631 C3FB4I 44303721 Ki > 470000 nM T84631 CQLA16 44303733 Ki = 104000 nM T84631 C5RZL0 44303743 Ki = 1700 nM T84631 CTE75P 44303769 Ki = 37000 nM T84631 C16GOI 44303778 Ki = 2800 nM T84631 C26ZUK 44303789 Ki = 5200 nM T84631 CN6V9A 44303803 Ki = 2300 nM T84631 C67ZRW 44303804 Ki = 188000 nM T84631 CB38WA 44303805 Ki = 12000 nM T84631 CL0U1A 44303806 Ki = 5700 nM T84631 CVO2D9 44303808 Ki = 99000 nM T84631 C0JZY5 44303810 Ki = 15000 nM T84631 CFJ4W3 44303811 Ki = 9400 nM T84631 CE0R9A 44303824 Ki > 470000 nM T84631 C5YF7O 44303839 Ki > 470000 nM T84631 C2LY4T 44303843 Ki = 1000 nM T84631 C3HXW6 44303858 Ki = 78 nM T84631 CYW9S8 44303912 Ki = 240000 nM T84631 CIQZ37 44303925 Ki = 88000 nM T84631 CJN72A 44303933 Ki = 2100 nM T84631 CXCY31 44303935 Ki > 78000 nM T84631 C4SN8T 44304006 Ki > 470000 nM T84631 CL16JC 44304046 Ki > 470000 nM T84631 CAM6R0 44304047 Ki > 470000 nM T84631 CR4V0L 44304084 Ki = 68000 nM T84631 CG37DH 44304086 Ki = 235000 nM T84631 C7UJH1 44304087 Ki = 55000 nM T84631 CG0R8N 44304097 Ki = 13000 nM T84631 CJ80KE 44304098 Ki > 470000 nM T84631 CG8TI6 44304099 Ki > 470000 nM T84631 C9W8QC 44304100 Ki > 470000 nM T84631 CE31BF 44304104 Ki > 470000 nM T84631 C9XIO1 44304105 Ki > 470000 nM T84631 C83YIU 44304139 Ki = 151000 nM T84631 CP5S9K 44304192 Ki = 470000 nM T84631 CKD98A 44304353 Ki = 350000 nM T84631 CDNY01 44304666 IC50 > 11000 nM T84631 CU86PQ 44304683 IC50 > 11000 nM T84631 C2WER6 44304686 IC50 = 1800 nM T84631 C8FQD7 44304721 IC50 = 250 nM T84631 C9T0AL 44304783 IC50 = 9500 nM T84631 CV5X7Z 44304784 IC50 = 1300 nM T84631 C4C5QV 44304795 IC50 > 11000 nM T84631 CK30FU 44304796 IC50 = 5700 nM T84631 CJ9ZC7 44304847 IC50 = 1100 nM T84631 C0CVL6 44304925 IC50 = 1500 nM T84631 C6VMS3 44304940 IC50 = 220 nM T84631 CH5T1S 44304949 IC50 = 14 nM T84631 CH5KL1 44304966 IC50 = 190 nM T84631 CW2ND0 44304967 IC50 > 11000 nM T84631 CX68LN 44304970 IC50 = 1 nM T84631 CR92NX 44304975 IC50 = 78 nM T84631 C9FPX1 44304983 IC50 = 14 nM T84631 CSC71I 44305011 IC50 = 7 nM T84631 CI28LX 44305020 IC50 = 140 nM T84631 CC94HD 44305021 IC50 = 1500 nM T84631 C47VUA 44305033 IC50 = 2900 nM T84631 CX6HR3 44305497 IC50 = 36 nM T84631 C1TU6Q 44305498 IC50 > 11000 nM T84631 CGM7D3 44305549 IC50 = 530 nM T84631 CM6VI1 44305564 IC50 = 41 nM T84631 C85BPT 44305569 IC50 = 590 nM T84631 C2CUS5 44305576 IC50 = 27 nM T84631 C0B8EM 44305583 IC50 = 230 nM T84631 CNE75U 44305589 IC50 = 84 nM T84631 CJ5GZ8 44305595 IC50 = 3 nM T84631 CXSN91 44305596 IC50 = 270 nM T84631 C8RXZ9 44305609 IC50 = 230 nM T84631 CJ9P6T 44305616 IC50 = 24 nM T84631 C1F5ZJ 44305618 IC50 = 27 nM T84631 CR0F5Q 44305620 IC50 = 31 nM T84631 C8WPQ1 44305624 IC50 = 12 nM T84631 CN91ZP 44305641 IC50 = 67 nM T84631 CGQA30 44305642 IC50 = 640 nM T84631 CG2K9Z 44305652 IC50 = 7 nM T84631 CJSV68 44305653 IC50 = 7 nM T84631 C13RXM 44305655 IC50 = 5 nM T84631 CJ13QC 44305697 IC50 = 12 nM T84631 C9MS8B 44305700 IC50 = 70 nM T84631 C5OT9C 44305701 IC50 = 25 nM T84631 C0OGD3 44305702 IC50 = 10 nM T84631 CO1Y2P 44305705 IC50 = 57 nM T84631 C36BTK 44305707 IC50 = 1300 nM T84631 CNBM39 44305717 IC50 = 8 nM T84631 C4OA9H 44305740 IC50 = 37 nM T84631 CF9K6V 44305751 IC50 = 150 nM T84631 CK8OA9 44305755 IC50 = 14 nM T84631 CR1B5E 44305767 IC50 = 18 nM T84631 C8I2WA 44305768 IC50 = 240 nM T84631 C6D4WM 44305778 IC50 = 390 nM T84631 CPE2R8 44305779 IC50 = 64 nM T84631 CS1T4V 44305783 IC50 = 100 nM T84631 CP5Q9V 44305791 IC50 = 8 nM T84631 CD4K9F 44305792 IC50 = 11 nM T84631 CLI7J5 44305799 IC50 = 140 nM T84631 C09VHZ 44305800 IC50 = 11 nM T84631 CWDY81 44305841 IC50 = 29 nM T84631 CLP78H 44305852 IC50 = 8 nM T84631 CKCQ26 44305853 IC50 = 8 nM T84631 C09HMY 44305854 IC50 = 15 nM T84631 COS9P8 44305862 IC50 = 7 nM T84631 C4BXN1 44305898 IC50 = 19 nM T84631 C6X1UY 44305922 IC50 = 71 nM T84631 CWL6P8 44305926 IC50 = 90 nM T84631 C2OPT7 44305934 IC50 = 120 nM T84631 CZ67XS 44305943 IC50 = 160 nM T84631 C18LVJ 44305951 IC50 = 13 nM T84631 CL1RT7 44305959 IC50 = 11 nM T84631 C9OQ6V 44305961 IC50 = 9 nM T84631 CYD8Q6 44305962 IC50 = 430 nM T84631 C30CNB 44305966 IC50 = 240 nM T84631 CP0R6L 44305992 IC50 = 6 nM T84631 CWG3K9 44306043 IC50 = 30 nM T84631 C4EBA0 44306054 IC50 = 45 nM T84631 CG0V3Z 44306077 IC50 = 6 nM T84631 C2G0UZ 44306101 IC50 = 10 nM T84631 CMIB37 44306212 IC50 = 8 nM T84631 CN97SF 44310725 Ki = 1000 nM T84631 CKP5W7 44311564 IC50 > 1100 nM T84631 C6TQ7D 44312627 IC50 = 14 nM T84631 CTW03S 44312639 IC50 = 93 nM T84631 C18PFJ 44312776 IC50 = 6.3 nM T84631 CGS74O 44312851 IC50 = 6.4 nM T84631 CM5RQ6 44312966 IC50 = 2930 nM T84631 CGND24 44312967 IC50 = 0.99 nM T84631 CRN7I3 44313020 IC50 > 10000 nM T84631 C6G0NQ 44313284 IC50 = 227 nM T84631 CYQ4I0 44313285 IC50 = 4.4 nM T84631 C2D0JU 44313317 IC50 = 170 nM T84631 CU8S5P 44313405 IC50 = 12100 nM T84631 C1KQR4 44313688 Ki = 9 nM T84631 CUA30F 44313689 Ki = 84 nM T84631 C87HJP 44313722 IC50 = 590 nM T84631 C3H5RB 44313873 IC50 = 46.4 nM T84631 C8V3IH 44313932 IC50 = 6.6 nM T84631 C6VP5I 44314000 IC50 = 7.89 nM T84631 CT2ZD9 44314001 IC50 = 13.2 nM T84631 CFXW28 44314002 IC50 = 3.26 nM T84631 CM10DN 44314053 IC50 = 0.86 nM T84631 CCK1W8 44314117 IC50 = 0.78 nM T84631 CT1X8J 44314118 IC50 = 1.87 nM T84631 C5H6VU 44314181 IC50 = 2.13 nM T84631 CSTP54 44314265 IC50 = 7.63 nM T84631 CE6B9A 44314318 IC50 = 246 nM T84631 C9IN4E 44314967 IC50 = 2900 nM T84631 C97NYB 44317783 IC50 = 2500 nM T84631 C5AK3D 44317785 IC50 > 2500 nM T84631 CW2X9Z 44318052 IC50 = 2500 nM T84631 CK58VB 44318182 IC50 = 5.78 nM T84631 CND9J7 44319469 Ki = 50.12 nM T84631 CEZ84L 44320397 IC50 = 28.9 nM T84631 CSK62O 44320493 IC50 = 49 nM T84631 CYT2Q4 44320495 IC50 = 7.2 nM T84631 CG36WH 44320752 IC50 = 3.6 nM T84631 CQ64CD 44320839 IC50 = 26.7 nM T84631 CK1EZ2 44320862 IC50 = 7.3 nM T84631 C7AMH4 44320876 IC50 = 20.6 nM T84631 CX73RG 44324726 Ki = 800 nM T84631 CMZ05T 44324727 Ki = 4900 nM T84631 CI5BY6 44324744 Ki = 7500 nM T84631 CKDN47 44324745 Ki = 2500 nM T84631 CWN4P7 44325526 Ki = 490 nM T84631 C1MT8R 44325527 Ki = 420 nM T84631 C1K5OT 44325647 Ki ~ 75 nM T84631 CG6ZC8 44325794 Ki = 36 nM T84631 CBD24R 44325803 Ki = 0.04 nM T84631 CZW79L 44325865 Ki = 240 nM T84631 C4Q8AC 44325938 Ki = 480 nM T84631 C61VAC 44325939 Ki = 510 nM T84631 CK92AD 44325940 Ki = 200 nM T84631 C6LWG3 44325946 Ki = 2470 nM T84631 C5TLH0 44325953 Ki = 720 nM T84631 CHI47Q 44325959 Ki = 240 nM T84631 C1DES8 44325967 Ki = 160 nM T84631 C5CLJ1 44325971 Ki = 28 nM T84631 CYOQ97 44325982 Ki > 1200 nM T84631 C3A2IO 44325983 Ki = 110 nM T84631 CZ9J5R 44326160 Ki = 1310 nM T84631 CO2F4Z 44326181 Ki = 380 nM T84631 CF92WZ 44326243 Ki = 37 nM T84631 CE8W2L 44326303 Ki = 3690 nM T84631 CK1EF5 44326322 Ki = 7050 nM T84631 C90VZO 44326339 Ki = 23 nM T84631 CXDN72 44326446 Ki = 2384 nM T84631 C3NCW0 44327306 Ki = 950 nM T84631 CFV5D6 44327462 Ki = 1700 nM T84631 CI56QW 44327465 Ki = 1400 nM T84631 CTDM97 44327484 Ki = 1800 nM T84631 C86YFO 44327490 Ki = 870 nM T84631 CE3UL6 44327872 Ki = 800 nM T84631 CSM3B6 44330879 IC50 = 34.8 nM T84631 CVM21A 44330906 IC50 = 635 nM T84631 CY72JW 44330907 IC50 = 34.8 nM T84631 CA4Y1P 44330934 IC50 = 1440 nM T84631 C3K6JA 44330969 IC50 = 23 nM T84631 CXW57P 44330970 IC50 = 25 nM T84631 CU9Z4M 44330999 IC50 = 7.8 nM T84631 C9KW3Q 44331002 IC50 = 842 nM T84631 CJ9Y8Z 44331003 IC50 = 55 nM T84631 C1X4UM 44331004 IC50 = 3450 nM T84631 C2SK9N 44331021 IC50 = 130 nM T84631 C2CS3N 44331022 IC50 = 640 nM T84631 CAB5T7 44331052 IC50 = 45 nM T84631 CR7F8L 44331114 IC50 = 31.3 nM T84631 C4NP5G 44331140 IC50 = 676 nM T84631 CSDQ73 44331145 IC50 = 2770 nM T84631 C4CJ5M 44331146 IC50 > 10000 nM T84631 CFK17Y 44331147 IC50 = 1780 nM T84631 C2BS5N 44331180 IC50 = 96.7 nM T84631 C1NR3B 44331189 IC50 = 10000 nM T84631 CF13OL 44331190 IC50 = 644 nM T84631 CE69GW 44331194 IC50 = 3 nM T84631 C3SU1R 44331210 IC50 = 762 nM T84631 CW5S8K 44332563 IC50 = 750 nM T84631 CB3XG7 44332586 IC50 = 490 nM T84631 C0WEP3 44332603 IC50 = 1590 nM T84631 CN5Q6W 44332607 IC50 = 1180 nM T84631 C9ECP7 44332620 IC50 = 5910 nM T84631 CKZ57W 44332622 IC50 = 420 nM T84631 C37XNC 44332629 IC50 = 440 nM T84631 CKJ49D 44332675 IC50 = 253 nM T84631 CQ7SG4 44332689 IC50 = 1 nM T84631 CNK6Z7 44332698 IC50 = 890 nM T84631 CZA7S5 44332713 IC50 = 3790 nM T84631 C89GTH 44332752 IC50 = 1610 nM T84631 CXO92K 44332753 IC50 = 890 nM T84631 CXUK98 44332765 IC50 = 110 nM T84631 CZ64UF 44332770 IC50 = 57 nM T84631 CA1IJ0 44332771 IC50 = 41 nM T84631 C5M2LB 44333833 Ki = 5000 nM T84631 CYNL31 44333951 Ki = 80 nM T84631 C0FE1Y 44333960 Ki = 1390 nM T84631 CJ2IM6 44333972 Ki = 22 nM T84631 CNF52U 44333992 Ki = 438 nM T84631 CIO79X 44334002 Ki = 320 nM T84631 CTUX56 44334003 Ki = 130 nM T84631 CS5X8Z 44334242 Ki = 46 nM T84631 CYX2N3 44334264 Ki = 99 nM T84631 CNTU54 44334314 Ki = 62 nM T84631 CDMP53 44334315 Ki = 15 nM T84631 CI3CT4 44334316 Ki = 392 nM T84631 CL05HM 44334318 Ki = 630 nM T84631 CN4TX8 44334349 Ki = 300 nM T84631 CQA75Y 44334374 Ki = 54 nM T84631 CI0C4V 44334382 Ki = 810 nM T84631 C0O1XG 44334554 Ki = 30 nM T84631 CHM49Q 44337735 Ki = 106000 nM T84631 CV7HW5 44337751 Ki = 92000 nM T84631 C39GBZ 44337785 Ki = 95000 nM T84631 CX35DM 44337794 Ki = 87300 nM T84631 CN1WI2 44337821 Ki = 90200 nM T84631 C61CGV 44337884 IC50 = 50 nM T84631 C4EFA8 44337894 IC50 = 210 nM T84631 C0HP3T 44337899 IC50 = 190000 nM T84631 CH0K1J 44337917 IC50 = 1400 nM T84631 CG6T9S 44337925 IC50 = 81000 nM T84631 CA10BE 44337935 IC50 = 20000 nM T84631 C4ATV2 44337945 IC50 = 1400 nM T84631 C2AN5G 44337986 IC50 = 69 nM T84631 CFH80Q 44337989 IC50 = 27000 nM T84631 CTD5Q8 44338012 IC50 = 33000 nM T84631 C5OVP7 44338032 IC50 = 31000 nM T84631 CI8U6O 44338109 IC50 = 698 nM T84631 CHX17O 44339365 Ki = 200000 nM T84631 CSA5H1 44339376 Ki = 179000 nM T84631 CZR56N 44339399 Ki = 69000 nM T84631 C9B0SQ 44339404 Ki = 228000 nM T84631 CC2K4G 44339417 Ki = 80000 nM T84631 C5WZ9O 44339442 Ki > 500000 nM T84631 C0G3LP 44339443 Ki = 81000 nM T84631 C4CZ2V 44339453 Ki > 200000 nM T84631 C7E4KL 44339464 Ki = 176400 nM T84631 CV53DA 44339470 Ki = 131000 nM T84631 CB6R0I 44339610 Ki = 370600 nM T84631 C7TOG2 44339650 Ki = 252000 nM T84631 CKA1T3 44341287 IC50 = 290 nM T84631 CZ9BF5 44341288 IC50 > 2500 nM T84631 C4XEK1 44341417 IC50 = 29.7 nM T84631 CXL2Q8 44341827 Ki = 149000 nM T84631 CQ2PR0 44342242 Ki = 26 nM T84631 CC0Z8V 44343581 IC50 = 6.1 nM T84631 CW76HT 44343582 IC50 = 15 nM T84631 CD0TW8 44343615 IC50 = 5 nM T84631 C9NZE1 44343799 IC50 = 0.7 nM T84631 CAIZ35 44343800 IC50 = 168.8 nM T84631 C0W6EI 44343845 IC50 = 311 nM T84631 C46IGW 44343852 IC50 = 312.5 nM T84631 C5H3NY 44343853 IC50 = 312.5 nM T84631 C7B5GK 44343857 IC50 > 2500 nM T84631 C40EHX 44343858 IC50 = 44.4 nM T84631 C91PVF 44343859 IC50 = 5.6 nM T84631 C4MS5Q 44343972 IC50 = 106 nM T84631 C3ZI7A 44343993 IC50 = 106 nM T84631 CMEI89 44343994 IC50 = 20.5 nM T84631 CEA17Z 44344039 IC50 = 346.3 nM T84631 CUO74X 44344054 IC50 = 10.6 nM T84631 C60GZW 44344100 IC50 = 10.6 nM T84631 CREZ48 44344153 IC50 = 79.1 nM T84631 CM2YO1 44345652 Ki = 900 nM T84631 CAY34C 44347478 Ki = 400000 nM T84631 CT0QN1 44347480 Ki > 1000000 nM T84631 CV6KA1 44347491 IC50 > 2500 nM T84631 C2EH3B 44347493 IC50 = 451 nM T84631 C65ORY 44347498 IC50 = 369 nM T84631 CN7L4W 44347532 IC50 = 627 nM T84631 C1UN9I 44347534 Ki = 370000 nM T84631 CM3P8Z 44347559 IC50 > 2500 nM T84631 CJ5A8E 44347561 IC50 > 2500 nM T84631 C0V2FL 44347624 Ki = 1000000 nM T84631 CTQ93K 44347853 Ki = 3.3 nM T84631 CA7C9J 44347854 Ki = 0.39 nM T84631 CE2SA3 44347864 IC50 = 470 nM T84631 CDMG63 44347916 Ki > 10000 nM T84631 CEP6C1 44347929 Ki > 10000 nM T84631 CC50UP 44347950 Ki > 10000 nM T84631 C0PR3S 44347951 Ki = 4600 nM T84631 CW2B1L 44347973 Ki > 10000 nM T84631 C7F6BG 44347997 Ki = 19 nM T84631 CKBN18 44348006 Ki > 10000 nM T84631 CX85LK 44348013 Ki > 10000 nM T84631 CQTB91 44348014 Ki = 6230 nM T84631 CXN6O9 44348021 Ki > 10000 nM T84631 C64JUL 44348030 Ki > 10000 nM T84631 C58MFB 44348077 IC50 = 5.6 nM T84631 C2AQR9 44348078 IC50 = 78 nM T84631 CJ1XO7 44348087 Ki = 8 nM T84631 C95OVC 44348092 Ki = 1.2 nM T84631 CQ8CK5 44348093 Ki = 13 nM T84631 CEL8P9 44348097 IC50 = 17 nM T84631 C31JWA 44348108 Ki = 5.4 nM T84631 CPV7C4 44348111 Ki > 10000 nM T84631 CO5Y7S 44348145 Ki > 10000 nM T84631 C6O8NQ 44348177 Ki > 10000 nM T84631 CQM0O4 44348226 Ki > 10000 nM T84631 CPD32J 44348228 Ki = 10700 nM T84631 CH61QP 44348436 IC50 = 8.4 nM T84631 CA74EQ 44348505 IC50 = 180 nM T84631 C2M6TU 44348587 IC50 = 32 nM T84631 CED0Q4 44348616 IC50 = 15 nM T84631 CZI93S 44348618 IC50 = 5900 nM T84631 CR68KY 44348619 IC50 = 41 nM T84631 C5H7ZW 44348620 IC50 = 63 nM T84631 C94NSH 44348621 IC50 = 980 nM T84631 CYS5G0 44348624 IC50 = 8.2 nM T84631 CFWR38 44348631 IC50 = 10 nM T84631 CV5F9W 44348635 IC50 = 7.6 nM T84631 C6QXM9 44348648 IC50 = 7 nM T84631 C04CQG 44348722 IC50 = 20 nM T84631 CBR0V8 44348733 IC50 = 440 nM T84631 CP2H0Q 44348745 IC50 = 1200 nM T84631 CT49QY 44351237 Ki = 12 nM T84631 CRY7N5 44351253 Ki = 1400 nM T84631 C2XC3I 44353392 IC50 = 28000 nM T84631 CE8S5Y 44353433 IC50 = 2800 nM T84631 C8WAB5 44353443 IC50 = 1500 nM T84631 C8BC3Z 44358436 Ki = 3900 nM T84631 CZA62D 44358571 Ki = 38000 nM T84631 CPO39C 44358576 Ki = 0.71 nM T84631 CI24PJ 44358733 Ki = 94 nM T84631 C4ZW0K 44359352 IC50 = 580 nM T84631 CVJ38H 44359353 IC50 = 1220 nM T84631 CB5T2W 44359354 IC50 = 460 nM T84631 CG0MW7 44359453 IC50 = 90 nM T84631 C1KL4Q 44359454 IC50 = 80 nM T84631 CMA5R7 44359487 IC50 = 1970 nM T84631 CZ9E1S 44359501 IC50 = 1130 nM T84631 CPU61I 44359598 IC50 = 390 nM T84631 CZ2T4O 44359609 IC50 = 4400 nM T84631 C6AFY1 44359621 IC50 = 600 nM T84631 C2Q1NY 44359626 IC50 = 360 nM T84631 C5GZ0D 44359648 IC50 = 1120 nM T84631 C82XKL 44359703 IC50 = 2500 nM T84631 C29ANK 44359723 IC50 = 2500 nM T84631 CQ5F0T 44359724 IC50 = 2500 nM T84631 C4Y5HK 44359726 IC50 = 2500 nM T84631 CIKY14 44359730 IC50 = 20.6 nM T84631 C40POZ 44359735 IC50 = 290 nM T84631 CF0V6J 44359754 IC50 = 2500 nM T84631 C5P3UG 44359755 IC50 = 2500 nM T84631 C5UKJ2 44359756 IC50 = 2500 nM T84631 CQ10VZ 44359794 IC50 = 2500 nM T84631 C5ES1X 44359805 IC50 = 1950 nM T84631 C5CTA0 44359810 IC50 = 471 nM T84631 CSV16F 44359885 IC50 > 2500 nM T84631 CD3R9Q 44359906 IC50 = 479 nM T84631 CMDB96 44360123 IC50 = 1100 nM T84631 C79GAF 44362167 Ki = 3499.45 nM T84631 C4Y0TJ 44362180 Ki = 34994.52 nM T84631 C3UYO8 44362181 Ki = 33113.11 nM T84631 CBFW89 44362183 Ki = 2301.44 nM T84631 CM4UL0 44362193 Ki = 25118.86 nM T84631 CA8B0F 44362198 Ki = 95499.26 nM T84631 CKY09S 44362201 Ki = 15995.58 nM T84631 CDM7W1 44362220 Ki = 39994.47 nM T84631 CH8S3E 44362221 Ki = 10964.78 nM T84631 CVY70U 44362237 Ki = 13001.7 nM T84631 CS6CA2 44362238 Ki = 2511.89 nM T84631 C7BEC4 44362239 Ki = 51999.6 nM T84631 C6W3XA 44362244 Ki = 70957.78 nM T84631 CK8PS0 44362245 Ki = 76032.63 nM T84631 CH5GN7 44362276 Ki = 15995.58 nM T84631 C7R6GJ 44362294 Ki = 57942.87 nM T84631 C47UOB 44362295 Ki = 41975.9 nM T84631 C9Y4GO 44362301 Ki = 79983.43 nM T84631 C8V2SK 44362302 Ki = 119949.93 nM T84631 CC8S0D 44362303 Ki = 77624.71 nM T84631 CH2JG8 44362312 Ki = 43351.09 nM T84631 C4OGX6 44362314 Ki = 76032.63 nM T84631 C7ZC4W 44362327 Ki = 16982.44 nM T84631 CL8FT9 44362329 Ki = 41495.4 nM T84631 C2BSP7 44362336 Ki = 26001.6 nM T84631 CO3T2F 44362337 Ki = 179887.09 nM T84631 C4DTY9 44362338 Ki = 2600.16 nM T84631 CVG80E 44362342 Ki = 17988.71 nM T84631 CL9CY2 44362343 Ki = 3198.9 nM T84631 C0D3TA 44362364 Ki = 2301.44 nM T84631 CW8BP5 44362367 Ki = 359749.34 nM T84631 CWZ91O 44362370 Ki = 17988.71 nM T84631 CR1W2C 44362374 Ki = 53951.06 nM T84631 CAR1I5 44362386 Ki = 26001.6 nM T84631 C3VU1F 44362388 Ki = 7603.26 nM T84631 CM43VS 44362389 Ki = 2511.89 nM T84631 C2JF6K 44362390 Ki = 46773.51 nM T84631 CC10SF 44362395 Ki = 38018.94 nM T84631 CC19SB 44362401 Ki = 64565.42 nM T84631 CC3LE4 44362404 Ki = 43651.58 nM T84631 CQ6HR5 44362406 Ki = 8090.96 nM T84631 CBP5C2 44362409 Ki = 100000 nM T84631 CFTC83 44362421 Ki = 35974.93 nM T84631 CE9I1R 44362422 Ki = 26977.39 nM T84631 C7GC4F 44362435 Ki = 19010.78 nM T84631 C2JPQ1 44362436 Ki = 8590.14 nM T84631 CIRJ69 44362445 Ki = 60255.96 nM T84631 C6IJ9O 44362457 Ki = 899.5 nM T84631 CG5X8L 44362464 Ki = 2197.86 nM T84631 CRZO54 44362466 Ki = 1513.56 nM T84631 C3UQ2G 44362474 Ki = 9705.1 nM T84631 CP7K9D 44362494 Ki = 46025.66 nM T84631 CNV52T 44362496 Ki = 16982.44 nM T84631 CZO9L1 44362497 Ki = 50003.45 nM T84631 CQM36L 44362517 Ki = 13001.7 nM T84631 CWVC27 44362544 Ki = 26977.39 nM T84631 CTXH42 44362558 Ki = 83176.38 nM T84631 CL5N9S 44362560 Ki = 21978.6 nM T84631 CD95NC 44362564 Ki = 7762.47 nM T84631 CG6MS9 44362581 Ki = 34994.52 nM T84631 CVR0L5 44362589 Ki = 130016.96 nM T84631 CA2PW9 44362609 Ki = 230144.18 nM T84631 C13XMI 44362611 Ki = 14125.38 nM T84631 CJD6N8 44362617 Ki = 10000 nM T84631 C3PWL5 44362648 Ki = 11994.99 nM T84631 C1N8AG 44362663 Ki = 21978.6 nM T84631 C74DSW 44362679 Ki = 6760.83 nM T84631 CX30CV 44362681 Ki = 19998.62 nM T84631 CSXG35 44362682 Ki = 109900.58 nM T84631 CC7TB6 44362760 Ki = 41020.41 nM T84631 CCAS16 44362802 Ki = 190107.83 nM T84631 C17REG 44362803 Ki = 1000000 nM T84631 CPF78Q 44362805 Ki = 639734.84 nM T84631 CJ6M0W 44362819 Ki = 3097.42 nM T84631 C2P6RJ 44364043 Ki = 200 nM T84631 C06RPS 44364101 Ki = 1000 nM T84631 C8H3IU 44364106 Ki = 200 nM T84631 C0B3TG 44364107 Ki = 80 nM T84631 CN46VL 44364123 Ki = 200 nM T84631 C1P0MS 44364177 Ki = 400 nM T84631 CYK89L 44364205 Ki = 3000 nM T84631 CP7K4W 44364302 Ki = 2000 nM T84631 C4LH6Q 44364310 Ki = 3000 nM T84631 CB85LE 44364311 Ki = 200 nM T84631 CDE32K 44364319 Ki = 30 nM T84631 CTC3O5 44364320 Ki = 2000 nM T84631 CSI3V9 44364329 Ki = 3000 nM T84631 CUM70S 44364371 Ki = 2000 nM T84631 C9Z7JD 44364382 Ki = 44 nM T84631 CT8QM1 44364445 Ki = 30 nM T84631 CTB86G 44364486 Ki = 55 nM T84631 C1ELX6 44364487 Ki = 1000 nM T84631 CQ1LM8 44364504 Ki = 100 nM T84631 CS2D1R 44364505 Ki = 400 nM T84631 CQE3K8 44364506 Ki = 200 nM T84631 CT10GM 44364862 Ki = 7.1 nM T84631 CDIR32 44364938 Ki = 210 nM T84631 CL1O0R 44364939 Ki > 5000 nM T84631 CYD1M4 44364940 Ki = 78 nM T84631 CXD05A 44364941 Ki = 960 nM T84631 COJ03I 44364946 Ki > 5000 nM T84631 C5M2CT 44364948 Ki > 5000 nM T84631 CM87YB 44364952 Ki > 5000 nM T84631 CD93ET 44364982 Ki > 5000 nM T84631 CG4RV3 44364999 Ki > 500 nM T84631 CTVZ78 44365103 Ki > 5000 nM T84631 CNO4X7 44365111 Ki > 5000 nM T84631 CIDS76 44365112 Ki = 4700 nM T84631 C4OE2C 44365192 Ki > 5000 nM T84631 CEH1M4 44365200 Ki > 5000 nM T84631 CFZ2T9 44365277 Ki = 280 nM T84631 C3GA5J 44365287 Ki = 1400 nM T84631 CN4D2F 44365289 Ki > 5000 nM T84631 C5YT9W 44366105 Ki = 1 nM T84631 CT1F2W 44366339 Ki = 0.46 nM T84631 C0L3YP 44367992 IC50 = 1570 nM T84631 CRD97F 44368086 IC50 = 7 nM T84631 C0HVT6 44368087 IC50 = 3 nM T84631 COQ97A 44368088 IC50 = 9 nM T84631 CZY31U 44368261 IC50 = 14900 nM T84631 C4B9CA 44368277 IC50 = 1050 nM T84631 C01GQT 44368278 IC50 = 6920 nM T84631 CJ4O0M 44368282 IC50 > 10000 nM T84631 C67DWF 44368293 IC50 = 14 nM T84631 CGQA02 44368299 IC50 = 3 nM T84631 C78XDG 44368377 IC50 = 25 nM T84631 C1LST9 44368378 IC50 = 31 nM T84631 CH3E9V 44368542 IC50 = 4060 nM T84631 CC2F9Z 44368575 IC50 = 6 nM T84631 C6OF4C 44368576 IC50 = 0.8 nM T84631 C37ZDX 44368590 IC50 = 7000 nM T84631 CCN24M 44368609 IC50 = 934 nM T84631 CTPD09 44368610 IC50 = 3933 nM T84631 CBT5V7 44368623 IC50 = 7 nM T84631 C62DWQ 44368626 IC50 = 153 nM T84631 CR12CY 44368637 IC50 = 500 nM T84631 CM2CE0 44368638 IC50 = 191 nM T84631 CAGX61 44368877 Ki = 2100 nM T84631 C8ABU5 44368882 Ki = 1400 nM T84631 C3PHI0 44369086 Ki = 0.15 nM T84631 CWK6U8 44369271 Ki = 0.013 nM T84631 C1HBT5 44369288 Ki < 0.005 nM T84631 C6XB0Y 44371477 Ki = 2900 nM T84631 C3T0PF 44372395 Ki = 0.82 nM T84631 CAJ92B 44372499 Ki = 2.3 nM T84631 CI32UH 44372518 Ki = 0.4 nM T84631 C7I3HS 44372533 Ki = 0.2 nM T84631 CJE89V 44372620 Ki = 8.2 nM T84631 C39FZP 44372663 Ki = 15000 nM T84631 C9I0BE 44372667 Ki = 500 nM T84631 CQLA75 44372683 Ki = 100000 nM T84631 CKFN05 44372724 Ki > 1000000 nM T84631 CTD36H 44372738 Ki = 140000 nM T84631 CI6MQ5 44372778 Ki = 10600 nM T84631 CUVD59 44372831 Ki = 6 nM T84631 CBLZ18 44372833 Ki = 1.1 nM T84631 CFH41R 44372839 Ki = 2000 nM T84631 C9COY7 44372840 Ki > 1000000 nM T84631 C34AWY 44372863 Ki = 140000 nM T84631 CZE15A 44372864 Ki = 28000 nM T84631 C7X5BE 44372865 Ki = 2000 nM T84631 C2E6TP 44372889 Ki = 28000 nM T84631 CNOV-41 44372899 Ki = 0.3 nM T84631 C36XWM 44372903 Ki = 410 nM T84631 C01VKC 44374066 Ki = 0.8 nM T84631 C3MX0H 44374677 Ki = 2.3 nM T84631 C4HSA0 44374690 Ki = 1.8 nM T84631 C2Y0SC 44375908 IC50 = 24000 nM T84631 C3C2XE 44375967 IC50 = 69 nM T84631 C69QAS 44375986 IC50 = 2 nM T84631 C34XTM 44375987 Ki = 0.013 nM T84631 CZVP71 44376028 IC50 = 1 nM T84631 CZA1N6 44376029 IC50 = 0.7 nM T84631 C58WMI 44376046 IC50 = 3 nM T84631 C74KVW 44376051 IC50 = 17 nM T84631 C6SC3T 44376056 IC50 = 771 nM T84631 C2NHP9 44376074 IC50 = 2 nM T84631 CE9N6S 44376077 IC50 = 21 nM T84631 C6QTS8 44376079 IC50 = 8 nM T84631 CEKQ15 44376084 IC50 = 0.62 nM T84631 C9T2QI 44376089 IC50 = 3 nM T84631 CD0W7C 44376100 IC50 = 2 nM T84631 CG78SI 44376101 IC50 = 320 nM T84631 CG9KH1 44376121 IC50 = 118 nM T84631 C23ZRU 44376219 IC50 = 510 nM T84631 C5PH2E 44376249 IC50 = 58 nM T84631 C0Y8QD 44376252 IC50 = 0.79 nM T84631 CD03ZI 44376253 IC50 = 38 nM T84631 CX98EC 44376254 IC50 = 85 nM T84631 C1F2JZ 44376255 IC50 = 116 nM T84631 C0MS6T 44376257 IC50 = 2 nM T84631 C7BS3N 44376258 IC50 = 13 nM T84631 C63JEF 44376259 IC50 = 0.9 nM T84631 C0Z9CS 44376264 IC50 = 1 nM T84631 CSRZ57 44376273 IC50 = 10 nM T84631 CCY74M 44376286 IC50 = 6 nM T84631 CP9IY1 44376287 IC50 = 6 nM T84631 C0S9XG 44376288 IC50 = 10 nM T84631 COX13N 44376289 IC50 = 1 nM T84631 CNC7F4 44376290 IC50 = 32 nM T84631 C6X7UG 44376311 IC50 = 0.89 nM T84631 C4TGW5 44376318 IC50 = 4 nM T84631 C28ZIJ 44376322 IC50 = 37 nM T84631 C51GPZ 44376323 IC50 = 154 nM T84631 C5Y6JB 44376326 IC50 = 1 nM T84631 CA59MK 44376327 IC50 = 5 nM T84631 C5R2PM 44376328 Ki = 0.17 nM T84631 CTZR83 44376339 Ki = 800 nM T84631 CDM65F 44376342 IC50 = 4 nM T84631 C6R5AG 44376343 IC50 = 2 nM T84631 C8M2PZ 44376385 IC50 = 65 nM T84631 CH95MO 44376405 Ki = 33900 nM T84631 CB87VR 44376416 IC50 = 2 nM T84631 C5VDG0 44376417 IC50 = 2 nM T84631 C1S5KV 44376423 IC50 = 29 nM T84631 CG64YQ 44376426 Ki = 1.4 nM T84631 COAE61 44376427 IC50 = 5 nM T84631 CXEG05 44376429 IC50 = 459 nM T84631 CP7CO4 44376432 IC50 = 144 nM T84631 CKI3R7 44376454 Ki = 300 nM T84631 CT8KB1 44376468 IC50 = 22000 nM T84631 CI03DP 44376475 IC50 = 3 nM T84631 CUVH30 44376476 IC50 = 4 nM T84631 CSW71I 44376504 Ki = 850 nM T84631 C7WTQ1 44376505 Ki = 7800 nM T84631 C9SW1H 44376514 IC50 = 11 nM T84631 CM75ZP 44376515 IC50 = 31 nM T84631 C51GQP 44376523 Ki = 910 nM T84631 CA7GW4 44376525 Ki = 500 nM T84631 CHW87S 44376544 IC50 = 7 nM T84631 CKHG50 44376548 Ki = 2300 nM T84631 CZ68PY 44376566 Ki = 2500 nM T84631 C3DLJ9 44376572 IC50 = 32 nM T84631 C41SQG 44376585 Ki = 10500 nM T84631 C1PK0O 44376651 Ki = 16 nM T84631 CXG42V 44376671 Ki = 6600 nM T84631 CJBO94 44376700 IC50 = 21 nM T84631 C3K7NA 44376701 IC50 = 3 nM T84631 CKSV26 44376702 IC50 = 13 nM T84631 CXZP98 44376712 Ki = 282 nM T84631 CUFO93 44376713 Ki = 120 nM T84631 C1Z3BF 44376731 IC50 = 11 nM T84631 CEKG07 44376754 Ki = 30 nM T84631 CQX98K 44376755 Ki = 28 nM T84631 C2JKH1 44376756 Ki = 42 nM T84631 CITM85 44376766 Ki = 25700 nM T84631 CV7I3K 44376788 Ki = 500 nM T84631 CV5J1M 44376828 Ki = 38000 nM T84631 C8P5YZ 44376949 IC50 = 6 nM T84631 C4XJD0 44377015 IC50 = 888 nM T84631 CQB2G9 44377016 IC50 = 370 nM T84631 C6QG0C 44377053 Ki = 100 nM T84631 C6A7VL 44377057 Ki = 145 nM T84631 CZ6W0S 44377280 Ki > 338 nM T84631 CVS76R 44377281 Ki = 49.2 nM T84631 CI2GS0 44377287 IC50 = 0.94 nM T84631 CKX32Z 44377301 Ki > 338 nM T84631 C7W2GD 44377304 IC50 = 1.08 nM T84631 C6RA4Q 44377310 Ki > 338 nM T84631 CG0S9N 44377311 Ki = 52.7 nM T84631 CP0V6X 44377320 IC50 = 2.2 nM T84631 C4KSG5 44377322 IC50 = 0.9 nM T84631 CH1NM4 44377327 Ki = 23 nM T84631 CTP28F 44377331 IC50 = 1.1 nM T84631 CN42TW 44377336 Ki > 338 nM T84631 CPE23W 44377369 Ki > 338 nM T84631 C30VGP 44377425 IC50 = 0.9 nM T84631 C39PST 44377471 Ki = 93 nM T84631 C5Q1LA 44377475 Ki > 338 nM T84631 CVHL28 44377478 Ki = 40 nM T84631 CT0G2D 44377544 Ki = 16 nM T84631 CK6I3F 44377546 IC50 = 2.6 nM T84631 CNUL43 44377548 IC50 = 4.3 nM T84631 CZBJ51 44377550 IC50 = 5.3 nM T84631 CHU5T4 44377558 IC50 = 2.1 nM T84631 CU49MW 44377570 Ki > 338 nM T84631 C1TVZ9 44377573 Ki > 338 nM T84631 C3LE7S 44377608 Ki > 338 nM T84631 C7Y4QI 44377622 Ki = 315 nM T84631 CXLT41 44377644 Ki > 338 nM T84631 CO7N6Y 44378546 Ki = 57600 nM T84631 CLXH02 44378887 Ki = 111000 nM T84631 CC4MP1 44380667 Ki > 6000 nM T84631 C5XC2T 44381273 Ki = 17000 nM T84631 CJ6M5B 44382389 IC50 = 2500 nM T84631 CTF4N6 44382391 IC50 = 2500 nM T84631 CAI65F 44382441 IC50 > 2500 nM T84631 CB5J9R 44383041 Ki >> 1200 nM T84631 C6LH5V 44383081 IC50 = 2500 nM T84631 C9SD3E 44383242 Ki = 10 nM T84631 CFN18Q 44383278 Ki >> 1200 nM T84631 C2Y8NB 44383311 Ki = 40 nM T84631 C2NG7K 44383318 Ki >> 1200 nM T84631 CL5D3K 44383321 Ki = 120 nM T84631 CTNC21 44383351 Ki > 1200 nM T84631 C5PW9E 44383425 IC50 > 2500 nM T84631 CLQ19H 44383460 Ki = 1200 nM T84631 C43KTU 44383519 Ki = 24 nM T84631 CNBG48 44383542 IC50 > 2500 nM T84631 C2IX5U 44383543 IC50 = 2360 nM T84631 C4YS2W 44383629 Ki = 390 nM T84631 CX8CZ4 44383764 Ki = 1200 nM T84631 CKOW56 44383765 Ki >> 1200 nM T84631 CJH1T9 44383975 Ki >> 1200 nM T84631 CL5HW0 44383976 Ki >> 1200 nM T84631 C5CF2Z 44383985 Ki = 1200 nM T84631 CG8V5P 44384040 Ki = 290 nM T84631 CTLY83 44384041 Ki = 17 nM T84631 CS0IP4 44384198 Ki = 0.8 nM T84631 C6IX3V 44384674 Ki = 30 nM T84631 CP74XU 44384744 Ki = 80 nM T84631 CGI1H8 44384745 Ki = 370 nM T84631 CHK87Y 44384746 Ki = 0.46 nM T84631 CR2VG0 44384747 Ki = 0.3 nM T84631 CUR5K2 44384798 Ki = 3.6 nM T84631 CQ1D0K 44384799 Ki = 5.9 nM T84631 CVYI62 44385066 Ki = 1.3 nM T84631 CJ01YE 44385090 Ki = 20 nM T84631 CV4N1P 44385091 Ki = 3.5 nM T84631 C1ZV8A 44385092 Ki = 0.6 nM T84631 COQ8S6 44385134 Ki = 22 nM T84631 CVGJ91 44385135 Ki = 417 nM T84631 CLWT03 44385136 Ki = 300 nM T84631 CT42KF 44385150 Ki = 3 nM T84631 CALR98 44385151 Ki = 1.1 nM T84631 CNH87R 44385152 Ki = 420 nM T84631 C43MAX 44385153 Ki = 300 nM T84631 CDT45B 44385195 Ki = 0.23 nM T84631 C7U0HZ 44385205 Ki = 4.6 nM T84631 CTX13E 44385259 Ki = 1050 nM T84631 CI91SG 44385260 Ki = 6 nM T84631 C4RV6U 44385263 Ki = 5 nM T84631 CNMA50 44385268 Ki = 370 nM T84631 C3DF2V 44385269 Ki = 80 nM T84631 C9Z1OC 44385301 Ki = 0.12 nM T84631 CHPL94 44385310 Ki = 840 nM T84631 C6VZ5Y 44385361 Ki = 340 nM T84631 CCR46P 44385364 Ki = 6.3 nM T84631 CPV5B7 44385418 Ki = 190 nM T84631 C8CE6A 44385432 Ki = 160 nM T84631 C56GNK 44385447 Ki = 0.8 nM T84631 CR47ZA 44385448 IC50 = 32 nM T84631 CG35IX 44385449 Ki = 1.8 nM T84631 C1QOM8 44385484 IC50 = 1.3 nM T84631 CG7LT1 44385488 IC50 = 53 nM T84631 C7B5NP 44385500 Ki = 0.1 nM T84631 C94GZU 44385541 IC50 = 76 nM T84631 CQ7G9I 44385552 Ki = 0.1 nM T84631 CUQ30E 44385556 IC50 = 23 nM T84631 CH0EJ5 44385561 Ki = 0.9 nM T84631 CZ9KO4 44385566 IC50 = 16 nM T84631 C3T9XK 44385607 IC50 = 6.3 nM T84631 CKY0P4 44385611 IC50 = 3.8 nM T84631 C8MF3J 44385614 IC50 = 39 nM T84631 CUS20V 44385673 IC50 = 40 nM T84631 CZ8XL6 44385679 Ki = 0.5 nM T84631 CL5BA4 44385729 Ki = 0.3 nM T84631 CQ1CH4 44385753 Ki = 0.7 nM T84631 C3DSN7 44385768 IC50 = 30 nM T84631 C8USN9 44385769 IC50 = 552 nM T84631 C2E8DS 44385771 IC50 = 10 nM T84631 C2VFC6 44385772 IC50 = 1.5 nM T84631 CN8V0W 44385779 IC50 = 2 nM T84631 CO2K6D 44385783 IC50 = 2.8 nM T84631 CIHV71 44385786 Ki = 2.8 nM T84631 CPOS98 44385789 Ki = 4.5 nM T84631 C2WYO3 44385799 Ki = 2.9 nM T84631 CJ5B9H 44385803 Ki = 30 nM T84631 C7ZNB9 44385807 IC50 = 66 nM T84631 CBEA65 44385842 IC50 = 0.8 nM T84631 CN5Q1G 44385864 Ki = 2 nM T84631 C4XY8T 44385865 Ki = 60 nM T84631 CC9M7E 44385869 IC50 = 136 nM T84631 C8WK4A 44385891 IC50 = 1.1 nM T84631 C3VSU7 44385892 IC50 = 1.8 nM T84631 C8T1ZD 44385893 Ki = 0.012 nM T84631 CY81KI 44385894 IC50 = 7 nM T84631 C42JCS 44385915 Ki = 2 nM T84631 C9F6LP 44385922 IC50 = 9.5 nM T84631 C37ZQR 44385924 Ki = 1.8 nM T84631 C3D2CL 44385935 Ki = 1.3 nM T84631 CUAY63 44385953 Ki = 1 nM T84631 CX1C3I 44385963 Ki = 3.3 nM T84631 CFPH43 44385967 Ki = 4 nM T84631 CW08OY 44385998 Ki = 0.2 nM T84631 CV6KG4 44386059 Ki = 0.1 nM T84631 CWR4Q6 44386101 Ki = 6.2 nM T84631 CJ48AC 44386102 Ki = 1 nM T84631 CV13WD 44386116 Ki = 0.3 nM T84631 CGU69V 44386179 IC50 = 6.9 nM T84631 CS65LH 44386185 IC50 = 230 nM T84631 CU0P5T 44386242 IC50 = 6.8 nM T84631 CU9J0D 44386250 IC50 = 171 nM T84631 C7NF2L 44386266 IC50 = 60 nM T84631 C0Z3LF 44386268 IC50 = 22 nM T84631 C9G7QW 44386322 IC50 = 156 nM T84631 C31CUG 44386326 IC50 = 11 nM T84631 CX58AM 44386358 Ki = 0.23 nM T84631 C2WCE4 44386371 IC50 = 176 nM T84631 CDR14L 44386384 IC50 = 3.5 nM T84631 C52POK 44386417 IC50 = 12 nM T84631 CRX1I9 44386418 IC50 = 35 nM T84631 CI23WQ 44386419 Ki = 0.2 nM T84631 CFQV46 44386424 IC50 = 74 nM T84631 CIBD76 44386484 IC50 = 82 nM T84631 C8ME4O 44386493 IC50 = 5.8 nM T84631 CD4AH3 44386540 IC50 = 2.3 nM T84631 CHAO48 44386542 IC50 = 15 nM T84631 C2D6XI 44386633 IC50 = 4.1 nM T84631 CLNO15 44386637 IC50 = 35 nM T84631 C81IMH 44386642 IC50 = 40 nM T84631 C8SYK9 44386783 Ki = 210000 nM T84631 C4JB0M 44386841 IC50 = 1.3 nM T84631 CJC27L 44386868 IC50 = 5.3 nM T84631 C5FI9N 44386929 IC50 = 2.8 nM T84631 C5MR1F 44386934 Ki = 0.6 nM T84631 C8K5HM 44387041 IC50 = 2.3 nM T84631 CA45DZ 44387044 IC50 = 3.6 nM T84631 C7IG6P 44387096 IC50 = 4.1 nM T84631 C07CMU 44387102 IC50 = 1.9 nM T84631 C39LUW 44387104 IC50 = 5 nM T84631 CK0A4V 44387120 Ki = 1 nM T84631 CJ9ED7 44387165 Ki = 0.2 nM T84631 C2QD1K 44387206 IC50 = 1.4 nM T84631 C6SV1C 44387258 IC50 = 38000 nM T84631 CN2GR5 44390800 Ki = 12400 nM T84631 CW3G5V 44390801 Ki = 19000 nM T84631 CESM50 44392171 Ki = 270 nM T84631 CRYN03 44392172 Ki = 300 nM T84631 C9FUI3 44392182 Ki > 180 nM T84631 CT1AO2 44392186 Ki = 90 nM T84631 CG8V4B 44392189 Ki > 9000 nM T84631 CVK58T 44392197 Ki = 130 nM T84631 C4CU6F 44392199 Ki = 65 nM T84631 C1K6IY 44392201 Ki > 9000 nM T84631 CKO0E4 44392205 Ki = 530 nM T84631 CAE80C 44392206 Ki = 270 nM T84631 CJC84M 44392224 Ki > 9000 nM T84631 CP1CF2 44392233 Ki = 200 nM T84631 CHQG45 44392249 Ki = 19 nM T84631 C45EDM 44392250 Ki = 120 nM T84631 CLM10G 44393633 IC50 = 300 nM T84631 COS35W 44393635 IC50 = 2000 nM T84631 C54IJH 44393646 IC50 = 30 nM T84631 C4J5YZ 44393648 IC50 = 30 nM T84631 C7F1EZ 44393650 IC50 = 200 nM T84631 CM15TG 44393671 IC50 = 200 nM T84631 CW2B4G 44393673 IC50 = 200 nM T84631 CAYT14 44393675 IC50 = 6 nM T84631 CI7OZ9 44393679 IC50 = 100 nM T84631 CO3B6P 44393688 IC50 = 400 nM T84631 C5BWQ3 44393690 IC50 = 100 nM T84631 CW7T2D 44393692 IC50 = 60 nM T84631 CD0O9Q 44393694 IC50 = 100 nM T84631 CU47SD 44393720 IC50 = 3000 nM T84631 C2Q6CA 44393722 IC50 = 40 nM T84631 C95LDV 44393724 IC50 = 300 nM T84631 CUFO09 44395404 Ki = 0.19 nM T84631 CJ45KG 44395699 IC50 = 11000 nM T84631 CN04TX 44395725 IC50 = 26000 nM T84631 CN7Y2C 44395728 IC50 = 12000 nM T84631 C81TGP 44395751 IC50 = 29000 nM T84631 CS7UY1 44395771 IC50 = 29000 nM T84631 COD05Q 44395835 IC50 = 13000 nM T84631 CA0ZU3 44395871 IC50 = 10000 nM T84631 C1G7ZQ 44395885 IC50 = 14000 nM T84631 CIB17E 44395901 IC50 = 22000 nM T84631 C4SUD5 44396124 IC50 = 59000 nM T84631 CCL3J1 44396183 IC50 = 12000 nM T84631 CEC5X2 44396195 IC50 = 20000 nM T84631 C9P1FN 44398617 Ki = 25 nM T84631 CD5SQ2 44398699 Ki = 3 nM T84631 CQH41I 44398720 Ki = 0.1 nM T84631 CE5S0J 44400525 IC50 = 1130 nM T84631 CB0N5T 44400527 Ki = 19 nM T84631 CH9TP3 44402039 Ki = 512 nM T84631 C49CME 44402191 Ki = 137 nM T84631 CL80DH 44402364 Ki = 417 nM T84631 CQ4J2A 44402383 Ki = 264 nM T84631 C8WR3I 44402428 Ki = 111 nM T84631 CJQ8X6 44402429 Ki = 104 nM T84631 C6CZ8H 44402442 Ki = 136 nM T84631 CPLF17 44402521 Ki = 442 nM T84631 C5JK1T 44402528 Ki = 731 nM T84631 C9CWT3 44402591 Ki = 40 nM T84631 CV0S6N 44402617 Ki = 632 nM T84631 C0EWM8 44402974 IC50 < 10000 nM T84631 CD16XV 44402976 IC50 = 51000 nM T84631 C90VXC 44402978 IC50 = 4800 nM T84631 CPLH23 44402980 IC50 = 29000 nM T84631 C3T9OL 44402982 IC50 = 3300 nM T84631 C0Z2RO 44402984 IC50 = 11000 nM T84631 C27KPR 44402986 IC50 = 4500 nM T84631 CX90NG 44402988 IC50 = 9600 nM T84631 CQT09E 44402990 IC50 = 8000 nM T84631 C3P2QU 44402994 IC50 = 11000 nM T84631 C9E6KX 44402996 IC50 = 12000 nM T84631 C7QC1J 44402998 IC50 = 26000 nM T84631 C59QOU 44403000 IC50 = 17000 nM T84631 CF4IG0 44403002 IC50 = 11000 nM T84631 COW8T1 44403004 IC50 = 17000 nM T84631 CPU19J 44403006 IC50 = 4100 nM T84631 CW3HV4 44403010 IC50 = 4300 nM T84631 CFI1B8 44403012 IC50 = 20000 nM T84631 C61JGY 44403016 IC50 = 59000 nM T84631 C7L6YO 44403018 IC50 = 5700 nM T84631 C8PE3F 44403020 IC50 = 13000 nM T84631 C7IP1V 44403898 IC50 = 120 nM T84631 CG5V0X 44403903 IC50 = 20 nM T84631 C4F8BL 44404188 Ki = 14 nM T84631 CB6JW0 44407541 Ki = 6 nM T84631 CZD4O6 44407546 Ki = 3 nM T84631 CJ7W6K 44407547 Ki = 3 nM T84631 C1G4BC 44407625 Ki = 46 nM T84631 CA6Q9U 44407762 Ki = 140 nM T84631 CK54BG 44407769 Ki = 80 nM T84631 CC9Z0M 44407770 Ki = 2 nM T84631 C8J5OE 44407777 Ki = 40 nM T84631 CP67EA 44411094 IC50 = 251 nM T84631 CM8OZ0 44411137 IC50 > 45000 nM T84631 C3BX5Y 44412781 Ki > 150000 nM T84631 CF5XO4 44413343 Ki = 3700 nM T84631 CTD42X 44413355 Ki = 1100 nM T84631 C9KQM2 44413356 Ki = 1300 nM T84631 CQDX92 44413619 Ki = 4600 nM T84631 C9S8YL 44413733 Ki = 13 nM T84631 CO8A0Y 44414333 Ki = 100000 nM T84631 CG6H0U 44415561 Ki = 30000 nM T84631 C3LCV6 44415581 Ki = 54000 nM T84631 CJ20PN 44416510 IC50 > 200000 nM T84631 CZK3N4 44416547 IC50 = 175400 nM T84631 CQA4B5 44416549 IC50 = 129000 nM T84631 CMVF02 44416571 IC50 = 43600 nM T84631 C3TJK6 44418750 IC50 = 14200 nM T84631 C9G1VL 44418752 IC50 = 14300 nM T84631 CHK10G 44418753 IC50 = 15400 nM T84631 C9OZ1M 44418754 IC50 > 20000 nM T84631 CRM0E4 44419084 IC50 = 2 nM T84631 C8LV0Y 44419092 IC50 < 0.5 nM T84631 CQ7PD9 44419104 IC50 = 0.7 nM T84631 CID32E 44419109 IC50 = 2 nM T84631 C54KZH 44419113 IC50 = 0.9 nM T84631 C18PXN 44419484 Ki = 0.04 nM T84631 CVJ85S 44421826 IC50 > 200000 nM T84631 CWVX31 44421837 IC50 > 200000 nM T84631 CD58ZY 44421845 IC50 > 200000 nM T84631 C48NZW 44426214 Ki = 0.32 nM T84631 COUZ56 44426215 Ki = 21 nM T84631 C3F2PN 44426216 Ki = 3900 nM T84631 CZ91LH 44426217 Ki = 3.3 nM T84631 CEV53U 44426218 Ki = 2.55 nM T84631 C8O6HV 44426219 Ki = 0.095 nM T84631 CJH6E4 44426220 Ki = 32 nM T84631 C3E2FT 44426221 Ki = 53 nM T84631 CW3G0D 44426222 Ki = 52 nM T84631 CN6VL5 44426224 Ki = 0.35 nM T84631 CG9XF0 44426226 Ki = 0.36 nM T84631 CQ7CF9 44426227 Ki = 3.4 nM T84631 CL4N6J 44426228 Ki = 0.76 nM T84631 CJ3B7D 44426229 Ki = 1.6 nM T84631 C5Q8HB 44426230 Ki = 4.9 nM T84631 C6RNO7 44426232 Ki = 4.9 nM T84631 CCGR09 44426234 Ki = 200 nM T84631 CD06OJ 44426235 Ki = 65 nM T84631 CR4D0U 44426236 Ki = 16 nM T84631 CIT7D5 44426237 Ki = 0.084 nM T84631 CW71LJ 44426238 Ki = 0.25 nM T84631 CY5Z6P 44426239 Ki = 0.059 nM T84631 CI0N7E 44426240 Ki = 0.24 nM T84631 C35VBM 44426241 Ki = 0.52 nM T84631 C0LIG6 44426243 Ki = 0.049 nM T84631 C9V2JR 44426244 Ki = 0.08 nM T84631 C72TBW 44426245 Ki = 0.87 nM T84631 CZ2GS7 44426246 Ki = 0.63 nM T84631 CPKM97 44426247 Ki = 1.7 nM T84631 C1MVS4 44426248 Ki = 0.92 nM T84631 C5W1RJ 44426249 Ki = 1 nM T84631 C8H5OR 44426250 Ki = 0.94 nM T84631 C8BE9L 44426251 Ki = 2.9 nM T84631 CT6C5J 44426252 Ki = 1.5 nM T84631 CCN6T9 44426253 Ki = 17 nM T84631 C1UYG6 44426254 Ki = 8.3 nM T84631 CGV1I0 44426657 IC50 = 40 nM T84631 CXI16J 44426658 IC50 = 50 nM T84631 CZ9O0J 44426660 IC50 > 30000 nM T84631 CJN3M1 44426799 IC50 > 30000 nM T84631 CO9Q4B 44427316 IC50 > 30000 nM T84631 CD9O6E 44427319 IC50 > 30000 nM T84631 C53IBP 44428362 Ki = 2.2 nM T84631 CI6QX0 44429068 IC50 = 90 nM T84631 CED2A3 44429069 IC50 > 100000 nM T84631 CG9DX2 44429071 IC50 > 100000 nM T84631 C58ODU 44429073 IC50 = 850 nM T84631 C9QB7L 44429075 IC50 = 950 nM T84631 CEP2S5 44429076 IC50 = 350 nM T84631 CP7AD2 44429077 IC50 = 250 nM T84631 CEQ2U3 44429078 IC50 = 49 nM T84631 C0OH9V 44429079 IC50 > 100000 nM T84631 CHE96M 44429080 IC50 = 1600 nM T84631 CNZF48 44429082 IC50 = 800 nM T84631 C1EGK3 44429083 IC50 = 170 nM T84631 CA6U4B 44429085 IC50 = 200 nM T84631 C4E3TU 44429087 IC50 = 1700 nM T84631 CRJ2G1 44429088 IC50 = 2300 nM T84631 CPT8U9 44429090 IC50 > 100000 nM T84631 CGHK29 44429092 IC50 > 100000 nM T84631 C2G5ZK 44429093 IC50 > 100000 nM T84631 CMWU43 44429094 IC50 = 560 nM T84631 CG7MW6 44429096 IC50 = 190 nM T84631 CS29AL 44429097 IC50 = 65 nM T84631 CWA2F9 44429098 IC50 = 100 nM T84631 CTUO84 44429099 IC50 = 39 nM T84631 CQS80V 44429101 IC50 = 58 nM T84631 C1Q0EO 44429102 IC50 = 11 nM T84631 CV7A9L 44429104 IC50 = 12 nM T84631 CL32QO 44429105 IC50 = 590 nM T84631 CB27IK 44429106 IC50 = 13 nM T84631 CH6Z7Y 44429108 IC50 = 8.1 nM T84631 C8IHX6 44429109 IC50 = 10 nM T84631 CO78JZ 44429110 IC50 = 13 nM T84631 C0PE1M 44432470 Ki = 1.7 nM T84631 CPER15 44432471 Ki = 3.2 nM T84631 CJO6Z9 44432472 Ki = 2.1 nM T84631 C3O9RC 44432473 Ki = 2.5 nM T84631 C4BSJ6 44432474 Ki = 10 nM T84631 C0D6SL 44432475 Ki = 1.3 nM T84631 CP2LI4 44432476 Ki = 3.9 nM T84631 CBAV03 44432477 Ki = 4.8 nM T84631 CN4QV7 44432489 Ki = 1 nM T84631 CE8NY0 44432490 Ki = 7.3 nM T84631 CZ20YU 44432491 Ki = 23 nM T84631 C3DK8P 44432494 Ki = 266 nM T84631 C5D3TL 44432495 Ki = 288 nM T84631 CF9Q5N 44432496 Ki = 27 nM T84631 CIH6B5 44432497 Ki = 36 nM T84631 CP84FK 44432498 Ki = 1220 nM T84631 C3YOB9 44432499 Ki = 7.92 nM T84631 CF8G5U 44432501 Ki = 170 nM T84631 C7BP9C 44432503 Ki = 124 nM T84631 CJ59VG 44432505 Ki = 1186 nM T84631 C8AJS7 44432506 Ki = 2610 nM T84631 C2M7XN 44432507 Ki = 138 nM T84631 C1YZ9P 44432508 Ki = 892 nM T84631 C14LPX 44432509 Ki = 226 nM T84631 C68JTP 44432510 Ki = 433 nM T84631 C8VC2O 44432511 Ki = 129 nM T84631 CAJ8R2 44432512 Ki = 360 nM T84631 CW0KC9 44432514 Ki = 603 nM T84631 C5LA6U 44432515 Ki = 7420 nM T84631 C2D5US 44432516 Ki = 8560 nM T84631 C05QPV 44432517 Ki = 14 nM T84631 CVX41Y 44432522 Ki = 37 nM T84631 C0BU8P 44432527 Ki = 0.94 nM T84631 C65WMJ 44432528 Ki = 4 nM T84631 CHC7Y5 44432529 Ki = 107 nM T84631 CO9E0L 44432534 Ki = 2.4 nM T84631 CXEL19 44432536 Ki = 0.44 nM T84631 CVO5Q1 44432538 Ki = 0.51 nM T84631 CMX28G 44432539 Ki = 0.95 nM T84631 CRO15T 44432542 Ki = 10 nM T84631 CEIG96 44432570 Ki = 82 nM T84631 C7L4YU 44432571 Ki = 11500 nM T84631 C4TO1Y 44432573 Ki = 4.2 nM T84631 CZ5WC2 44432574 Ki = 929 nM T84631 C0KJ7B 44432576 Ki = 1.3 nM T84631 CMP70C 44432577 Ki = 0.71 nM T84631 C4NWL3 44434801 Ki = 0.21 nM T84631 C90KHC 44434802 Ki = 0.84 nM T84631 CDI09P 44434803 Ki = 27 nM T84631 CYKG20 44434804 Ki = 7.9 nM T84631 CAB7R9 44434805 Ki = 10870 nM T84631 CHZ0U3 44434806 Ki = 1 nM T84631 CS6ZY1 44434807 Ki = 0.27 nM T84631 CR16BF 44434808 Ki = 0.56 nM T84631 CQIX73 44434809 Ki = 1.9 nM T84631 CFLI30 44434810 Ki = 2.1 nM T84631 C1GZT7 44434811 Ki = 1.6 nM T84631 C2TK5Q 44434812 Ki = 1.6 nM T84631 CM3T0U 44434813 Ki = 0.39 nM T84631 C4HL3O 44434814 Ki = 3 nM T84631 C5R8HJ 44434815 Ki = 2.6 nM T84631 CPA5X7 44434816 Ki = 2.6 nM T84631 C7FJR9 44434817 Ki = 18 nM T84631 COG34X 44434818 Ki = 0.58 nM T84631 CRW87S 44434819 Ki = 3.9 nM T84631 CZ27MI 44434820 Ki = 2.8 nM T84631 CAZ59V 44434822 Ki = 2 nM T84631 C27VMW 44434824 Ki = 1.3 nM T84631 C51RUQ 44434825 Ki = 1.7 nM T84631 CH2L5P 44434826 Ki = 2.1 nM T84631 C9JD8H 44434829 Ki = 2.2 nM T84631 CYHV92 44434830 Ki = 0.36 nM T84631 CT6XL4 44434831 Ki = 0.74 nM T84631 CWA82Q 44434833 Ki = 0.93 nM T84631 C7PF0V 44434834 Ki = 0.44 nM T84631 C9T1DP 44434835 Ki = 0.64 nM T84631 CE3R5S 44434836 Ki = 1.7 nM T84631 C2OCL7 44434838 Ki = 1.7 nM T84631 CY0Z4T 44434840 Ki = 0.56 nM T84631 C4ADI5 44435823 Ki = 2.3 nM T84631 C30CFX 44436704 IC50 > 10000 nM T84631 CLU2J3 44441275 IC50 = 270 nM T84631 CJ67AP 44441276 IC50 > 10000 nM T84631 CKJ61O 44441277 IC50 = 3200 nM T84631 C53IBS 44441278 IC50 > 10000 nM T84631 C5DKP6 44441279 IC50 = 4400 nM T84631 CBV16E 44441280 IC50 > 10000 nM T84631 C97RGS 44441281 IC50 > 10000 nM T84631 C1N8RW 44441282 IC50 = 265 nM T84631 C2ZO6L 44441283 IC50 = 2000 nM T84631 CHB06C 44441284 IC50 = 118 nM T84631 C8WL7U 44441285 IC50 = 86 nM T84631 C3BPD0 44441286 IC50 = 175 nM T84631 CVIO95 44441287 IC50 = 11.3 nM T84631 C0D1CR 44441288 IC50 > 1400 nM T84631 CIK8L7 44441289 IC50 > 10000 nM T84631 CB49OX 44441290 IC50 = 753 nM T84631 CS90XV 44443528 IC50 = 1100 nM T84631 C0IPW3 44443531 IC50 = 150 nM T84631 CV5CK0 44443532 IC50 = 18 nM T84631 CFW4B7 44443548 IC50 = 436 nM T84631 CD1WV5 44443552 IC50 = 70 nM T84631 C20ZPQ 44443557 IC50 = 61 nM T84631 CL7O4R 44443558 IC50 = 130 nM T84631 CL68HN 44443560 IC50 = 40 nM T84631 CW31AS 44443863 Ki = 4 nM T84631 CZTC23 44444412 Ki = 1400 nM T84631 CT0K6W 44444413 Ki = 0.82 nM T84631 C2GQ4X 44444414 Ki = 19 nM T84631 CG3IT9 44444415 Ki = 1 nM T84631 CN7U2V 44444416 Ki = 0.63 nM T84631 C5DHI1 44444417 Ki = 1400 nM T84631 C50JGC 44444418 Ki = 2.2 nM T84631 C5TG0M 44446364 Ki = 1.1 nM T84631 CX02SN 44446365 Ki = 0.7 nM T84631 CUN0M5 44446366 Ki = 8.9 nM T84631 C0NB1S 44446367 Ki = 2.7 nM T84631 CGC4U3 44446368 Ki = 4.4 nM T84631 CEQ3K7 44446375 Ki = 6.3 nM T84631 C90HMC 44446376 Ki = 15.5 nM T84631 C14UGA 44446377 Ki = 74.6 nM T84631 CDJH35 44446378 Ki = 215 nM T84631 CZ07YI 44446379 Ki = 80 nM T84631 C2H1ZM 44446380 Ki = 0.2 nM T84631 CS59RX 44446381 Ki = 0.1 nM T84631 CUT3E2 44446382 Ki = 2 nM T84631 CVQ2A5 44446383 Ki = 1.1 nM T84631 CQYA21 44446384 Ki = 6.2 nM T84631 CLX79F 44446385 Ki < 0.4 nM T84631 C63ALD 44446386 Ki < 0.3 nM T84631 C15NOL 44446387 Ki = 14 nM T84631 CHV7B9 44446388 Ki = 0.4 nM T84631 C1K3BV 44446389 Ki = 1.8 nM T84631 CZA52B 44446390 Ki = 11.8 nM T84631 C7AJ3M 44446391 Ki = 6 nM T84631 C7X4ZE 44446392 Ki = 9.1 nM T84631 CPB7H6 44446393 Ki = 180 nM T84631 C78RKU 44446394 Ki = 2334 nM T84631 CN8SC7 44446622 Ki = 1.5 nM T84631 CXT60W 44446625 Ki = 0.68 nM T84631 C8PW5C 44446626 Ki = 0.53 nM T84631 C2OX0A 44446627 Ki = 0.07 nM T84631 CGE82I 44446629 Ki = 0.16 nM T84631 CKJV95 44446630 Ki = 4.7 nM T84631 C4RVO9 44446632 Ki = 22 nM T84631 C4WFK6 44446634 Ki = 2.8 nM T84631 C1HOX5 44446638 Ki = 2.3 nM T84631 C5WH9G 44446642 Ki = 0.97 nM T84631 C47NBK 44446644 Ki = 0.57 nM T84631 CU3YD7 44446648 Ki = 0.32 nM T84631 CC9LB6 44446651 Ki = 0.34 nM T84631 CSR9L5 44446652 Ki = 12 nM T84631 CH27CY 44446654 Ki = 6.9 nM T84631 CNX71T 44446656 Ki = 3.3 nM T84631 C8T7LJ 44446659 Ki = 1 nM T84631 CVQN67 44449252 Ki = 0.14 nM T84631 CS0M1X 44449283 Ki = 0.45 nM T84631 C0ER8M 44449284 Ki = 2 nM T84631 CO06UN 44449312 Ki = 0.14 nM T84631 CH2KY6 44449344 Ki = 2.2 nM T84631 CM7Z2Y 44449346 Ki = 7670 nM T84631 CI19PT 44449347 Ki = 0.12 nM T84631 CO8DL4 44449376 Ki = 1.1 nM T84631 CTY1O5 44449377 Ki = 59 nM T84631 CX7VI4 44449404 Ki = 0.62 nM T84631 CM79OK 44449405 Ki = 0.21 nM T84631 CBT6Y9 44449406 Ki = 4.2 nM T84631 CW0K7B 44449442 Ki = 1560 nM T84631 CVQA35 44449443 Ki = 0.14 nM T84631 CT1EI5 44449445 Ki = 0.58 nM T84631 C5Y9CT 44449469 Ki = 43 nM T84631 C0JD6K 44449470 Ki = 1 nM T84631 CP23WS 44449471 Ki = 3 nM T84631 CQ0P1T 44449498 Ki = 1.2 nM T84631 CEN98O 44449697 Ki = 0.005 nM T84631 CLNS10 44449700 Ki = 0.24 nM T84631 C1ATS9 44449734 Ki = 0.065 nM T84631 C8IC1F 44449735 Ki = 0.047 nM T84631 C0Y6AD 44450537 IC50 = 12 nM T84631 C15UNI 44450551 IC50 = 35 nM T84631 CY6WC9 44450552 IC50 = 24 nM T84631 C04NRS 44450553 IC50 = 21 nM T84631 CV0LM3 44450559 IC50 = 29 nM T84631 CFWS94 44450560 IC50 = 24 nM T84631 CTU6D5 44450561 IC50 = 78 nM T84631 CF8KZ6 44450562 IC50 = 840 nM T84631 C6LQ5H 44450623 IC50 = 18 nM T84631 C6RP8L 44450625 IC50 = 22 nM T84631 CQC3K0 44450638 IC50 = 41 nM T84631 CSQ67W 44450639 IC50 = 45 nM T84631 CN12UB 44450640 IC50 = 87 nM T84631 C2RS0U 44450654 IC50 = 57 nM T84631 CKT83Q 44450655 IC50 = 20 nM T84631 CPM47O 44450667 IC50 = 18 nM T84631 CTI72P 44450668 IC50 = 93 nM T84631 CC6A4Y 44453083 IC50 = 110 nM T84631 C06BVN 44453135 IC50 = 21 nM T84631 C94URG 44453211 IC50 = 0.6 nM T84631 CCR38H 44453230 Ki = 0.43 nM T84631 C0L4EK 44453237 IC50 = 2700 nM T84631 CRZ3U1 44453240 IC50 = 2 nM T84631 C12TPH 44453241 IC50 = 2 nM T84631 C5Y7AL 44453264 Ki = 2.7 nM T84631 CVQ68S 44453294 Ki = 1.1 nM T84631 CCO3E0 44453323 Ki = 2.2 nM T84631 CUAC72 44453324 Ki = 0.84 nM T84631 C4D2EV 44453334 IC50 = 17 nM T84631 CU3BS5 44453335 IC50 = 4 nM T84631 C2SH5L 44453374 IC50 = 320 nM T84631 CSC10P 44453375 IC50 = 8 nM T84631 CHRV89 44453404 Ki = 2.3 nM T84631 CH13TZ 44453406 Ki = 2.2 nM T84631 C0U3TE 44453410 IC50 = 770 nM T84631 CDZJ38 44453414 IC50 = 2 nM T84631 CK3HE8 44453438 Ki = 3200 nM T84631 C0V3FO 44453445 IC50 = 3 nM T84631 CN65UR 44453506 IC50 = 380 nM T84631 CMQ7F1 44453531 Ki = 61 nM T84631 CMNY25 44453560 Ki = 160 nM T84631 C39RNM 44453561 Ki = 420 nM T84631 CVKT34 44453567 IC50 = 1 nM T84631 C6FI3U 44453568 IC50 = 44 nM T84631 C7KER6 44453580 Ki = 16 nM T84631 C0OK6W 44453582 Ki = 28 nM T84631 C6WGH0 44453588 IC50 = 85 nM T84631 CV7FC4 44453589 IC50 = 8 nM T84631 CBMH30 44453593 IC50 = 28 nM T84631 C7T9XG 44453617 Ki = 0.35 nM T84631 C67GMZ 44453618 Ki = 0.21 nM T84631 COC52H 44453619 Ki = 18 nM T84631 C7KD4P 44453642 Ki = 0.71 nM T84631 CB86HU 44453827 IC50 = 2 nM T84631 C1OX5F 44454953 IC50 = 7.8 nM T84631 C9K1OZ 44454955 IC50 = 8.4 nM T84631 CH08YV 44454956 IC50 = 5.6 nM T84631 CG07OV 44454984 IC50 = 9 nM T84631 CXD79F 44455009 IC50 = 9.3 nM T84631 CYPN89 44455011 IC50 = 110 nM T84631 CD81LJ 44455042 IC50 = 4.5 nM T84631 CMU0N2 44455044 IC50 = 45 nM T84631 C8ZMQ1 44455079 IC50 = 28 nM T84631 CUP8J7 44455081 IC50 = 48 nM T84631 C6OXL4 44455113 IC50 = 8.6 nM T84631 COKJ02 44455114 IC50 = 530 nM T84631 CQ4F1I 44455154 IC50 = 62 nM T84631 C1MU6Z 44455155 IC50 = 130 nM T84631 CBI54T 44455189 IC50 = 10 nM T84631 CV6K4Z 44455262 IC50 = 41 nM T84631 C36KNH 44455401 IC50 = 26 nM T84631 COM4K5 44455402 IC50 = 56 nM T84631 C7RV6S 44455427 IC50 = 47 nM T84631 CMJK06 44455903 Ki = 895 nM T84631 C3D6IN 44455904 Ki = 0.5 nM T84631 CUF96X 44455934 Ki < 0.3 nM T84631 C7R0VC 44455936 Ki = 5.9 nM T84631 C91XPS 44455972 Ki = 4.5 nM T84631 C8T6VP 44455976 Ki = 2.3 nM T84631 C94SCR 44456008 Ki = 0.6 nM T84631 CHB84J 44456009 Ki = 0.8 nM T84631 CRI4A1 44456042 Ki < 1 nM T84631 CJ0WH2 44456043 Ki = 3.1 nM T84631 CET18J 44456076 Ki = 0.2 nM T84631 C4JW5U 44456118 Ki = 0.2 nM T84631 CG82AV 44456315 Ki = 5 nM T84631 CVP6D1 44456316 Ki = 16.4 nM T84631 CN7I5U 44456317 Ki < 1 nM T84631 C2HYR5 44456355 Ki = 0.6 nM T84631 CB80FW 44456356 Ki = 0.4 nM T84631 CQ2LF9 44456386 Ki = 1.2 nM T84631 C3YT1F 44456387 Ki = 0.4 nM T84631 CZJ84G 44456388 Ki = 14.7 nM T84631 CONZ35 44456432 Ki = 14.7 nM T84631 CPX63S 44456433 Ki = 125 nM T84631 C8P7AO 44456477 Ki = 29.3 nM T84631 CEVH54 44456525 IC50 > 5000 nM T84631 C2T6FK 44456526 IC50 > 5000 nM T84631 CSJY82 44456652 IC50 = 37 nM T84631 CSA87I 44456653 IC50 = 95 nM T84631 CEX4F8 44456675 IC50 = 85 nM T84631 CA80WD 44456676 IC50 = 60 nM T84631 CSRK86 44456702 IC50 = 120 nM T84631 C42JQR 44456704 IC50 = 54 nM T84631 C96YAC 44456722 IC50 = 64 nM T84631 C1C0LS 44456751 IC50 = 250 nM T84631 CZ5Q1B 44456777 IC50 = 160 nM T84631 C4R1JB 44456779 IC50 = 720 nM T84631 CAIN46 44456806 IC50 = 140 nM T84631 CZ7D3W 44456807 IC50 = 840 nM T84631 CEC75K 44456850 IC50 = 470 nM T84631 CPYT84 44456869 IC50 > 5000 nM T84631 C1TFA0 44456897 IC50 > 5000 nM T84631 C6ERW2 44456898 IC50 = 720 nM T84631 C6TFX8 44457896 Ki = 54 nM T84631 C2VAB4 44457926 Ki = 200 nM T84631 CPXA19 44457985 Ki = 100 nM T84631 C3H9RE 44458036 Ki = 120 nM T84631 COE83M 44458061 Ki = 1.1 nM T84631 C0GCJ3 44458084 Ki = 5800 nM T84631 CB4P1V 44458141 Ki = 17 nM T84631 C3B0TA 44458142 Ki = 110 nM T84631 CWS61M 44458143 Ki = 120 nM T84631 C5Z9CS 44458144 Ki = 360 nM T84631 CA2ZK4 44458145 Ki = 120 nM T84631 C1DBQ3 44458182 Ki = 60 nM T84631 CS1TF7 44460215 IC50 > 2500 nM T84631 CH61KG 44460246 IC50 > 2500 nM T84631 CWB04E 44462312 IC50 = 43.2 nM T84631 CIO47G 44473069 IC50 = 10 nM T84631 CFL8D2 44473070 IC50 = 12 nM T84631 C7S5LI 44473071 IC50 = 24 nM T84631 C75XDR 44473072 IC50 = 17 nM T84631 C06IAS 44473073 IC50 = 32 nM T84631 CZ13SI 44473074 IC50 = 28 nM T84631 CY64AE 44473075 IC50 = 15 nM T84631 CM3S2V 44473076 IC50 = 6 nM T84631 CL18JO 44473077 IC50 = 7 nM T84631 CJ6A4T 44473078 IC50 = 5 nM T84631 CSV5O4 44473081 IC50 = 6 nM T84631 C28UIH 44473082 IC50 = 2 nM T84631 CYZV01 44473085 IC50 = 55 nM T84631 CC75ON 44473086 IC50 = 4 nM T84631 CA2P3T 44473087 IC50 = 3 nM T84631 C3H8CB 44473088 IC50 = 50 nM T84631 CH12VF 44473089 IC50 = 4 nM T84631 CYP8O4 44473090 IC50 = 6 nM T84631 CSR40D 44473091 IC50 = 9 nM T84631 CS0HV7 44473092 IC50 = 56 nM T84631 CUZ97H 44473093 IC50 = 10 nM T84631 CSFM32 44473094 IC50 = 17 nM T84631 C2OT5K 44473095 IC50 = 4 nM T84631 C4H0DY 44473096 IC50 = 5 nM T84631 C7S8OZ 44473097 IC50 = 3.3 nM T84631 CO19AD 44473098 IC50 = 12 nM T84631 CTP32R 44473099 IC50 = 6 nM T84631 CBRX82 44520907 IC50 = 120 nM T84631 CP4XV3 44520908 IC50 = 1100 nM T84631 CTC95U 44520909 IC50 = 1900 nM T84631 CB5IC4 44520910 IC50 = 2300 nM T84631 CRPO96 44520911 IC50 = 69 nM T84631 CN5AX7 44520912 IC50 = 55 nM T84631 CZ54XV 44520913 IC50 = 1.4 nM T84631 C2IN6J 44520914 IC50 = 49 nM T84631 C4CT6V 44520915 IC50 = 3.5 nM T84631 CJY68M 44520916 IC50 = 4.8 nM T84631 CLA7J5 44520917 IC50 = 5.7 nM T84631 CEI82S 44520918 IC50 = 15 nM T84631 CGC10V 44520919 IC50 = 3.2 nM T84631 CS38ZY 44520920 IC50 = 4000 nM T84631 COT9K1 44520921 IC50 = 3 nM T84631 C8SOG1 44520922 IC50 = 4.1 nM T84631 CBLG40 44520923 IC50 = 870 nM T84631 CPY9M7 44520924 IC50 = 35 nM T84631 CUJ6F0 44520925 IC50 = 12 nM T84631 CM9HL2 44520927 IC50 = 4.9 nM T84631 C1H2DQ 44520928 IC50 = 12 nM T84631 C4V5OJ 44520929 IC50 = 9.5 nM T84631 CY9IN4 44520930 IC50 = 3.4 nM T84631 CVZW52 44537923 IC50 = 2700 nM T84631 C0SR7G 44560382 Ki = 0.14 nM T84631 CFSV74 44560383 Ki = 1.4 nM T84631 CH8F6K 44560756 Ki = 0.038 nM T84631 C7AIN2 44560776 Ki = 2.4 nM T84631 CMG1Z3 44560812 Ki = 5.8 nM T84631 CGC65N 44560813 Ki = 30 nM T84631 C68JXO 44560836 Ki = 54 nM T84631 CM6PB1 44560883 Ki = 0.57 nM T84631 CZD69W 44560918 Ki = 0.042 nM T84631 C6SI5T 44565123 Ki = 25084 nM T84631 C1F8OZ 44565598 IC50 = 2 nM T84631 CT47ME 44565599 IC50 = 0.5 nM T84631 C6CE3S 44565600 IC50 = 0.5 nM T84631 CGR65Q 44565601 IC50 = 0.5 nM T84631 CC7KE3 44565602 IC50 = 1.2 nM T84631 C8L5HU 44565603 IC50 = 0.9 nM T84631 C41GHV 44565623 IC50 = 1.3 nM T84631 CW5EX0 44565624 IC50 = 1 nM T84631 CDG04W 44565625 IC50 = 1.2 nM T84631 C0XC6Y 44565626 IC50 = 1.2 nM T84631 COJE58 44565627 IC50 = 0.9 nM T84631 C7EF2R 44565628 IC50 = 3 nM T84631 CB7WF1 44565629 IC50 < 0.5 nM T84631 C0MHX6 44565630 IC50 = 3 nM T84631 C14HKO 44565631 IC50 = 0.5 nM T84631 CR09OH 44565632 IC50 = 0.4 nM T84631 CA0XT3 44565740 IC50 < 0.5 nM T84631 CY4HL8 44565741 IC50 = 1.5 nM T84631 CD94RJ 44565746 IC50 = 1.3 nM T84631 C2EJ4X 44565747 IC50 = 1.1 nM T84631 C9XT0W 44565748 IC50 = 3 nM T84631 C5NTH8 44565757 IC50 = 6 nM T84631 CXZK47 44565758 IC50 = 1.1 nM T84631 C48BCZ 44565759 IC50 = 7 nM T84631 CBV9Z6 44565760 IC50 = 2 nM T84631 C7MSE6 44565784 IC50 = 0.7 nM T84631 CAE2K6 44565785 IC50 = 1 nM T84631 CW4DZ0 44565786 IC50 = 3 nM T84631 C4O1MU 44565787 IC50 = 1 nM T84631 C9GXH4 44565788 IC50 = 6 nM T84631 CKF9Z4 44565789 IC50 = 17 nM T84631 C4CX2F 44565790 IC50 = 10 nM T84631 CEW6G1 44569299 Ki = 10 nM T84631 C9JNT3 44569300 Ki = 1700 nM T84631 C9XE7Q 44569301 Ki = 92000 nM T84631 CZI8D7 44569333 Ki = 430000 nM T84631 CR4CP6 44569359 Ki = 55000 nM T84631 C9JF7W 44569667 Ki = 4400 nM T84631 C61IJB 44569732 Ki = 8000 nM T84631 CR36MB 44569733 Ki = 61000 nM T84631 CE25UL 44569767 Ki = 20000 nM T84631 C0CZ4I 44569768 Ki = 14000 nM T84631 CIR4M0 44569769 Ki = 5400 nM T84631 C02SHD 44569811 Ki = 700 nM T84631 CG3LE9 44569812 Ki = 5600 nM T84631 CCU7V0 44569813 Ki = 910 nM T84631 C8BR6E 44569843 Ki = 660 nM T84631 C7Q9BH 44569844 Ki = 3400 nM T84631 CZ35OW 44569845 Ki = 420 nM T84631 CHV9C1 44569846 Ki = 630 nM T84631 C5JQ4W 44569889 Ki = 1600 nM T84631 CE1O4I 44569890 Ki = 3500 nM T84631 C4JU7I 44569891 Ki = 150 nM T84631 CGS83Z 44569892 Ki = 250 nM T84631 CFKJ12 44570705 IC50 = 4.5 nM T84631 CCA09Y 44570706 IC50 = 2.6 nM T84631 C7QWX9 44570769 IC50 = 2.9 nM T84631 C64OEB 44570770 IC50 = 2.3 nM T84631 C3KF1Y 44570771 IC50 = 3.5 nM T84631 CJVS07 44570772 IC50 = 2.5 nM T84631 C60XGS 44571089 IC50 = 3.4 nM T84631 C7DBF4 44571090 IC50 = 2.2 nM T84631 CGRP54 44571091 IC50 = 4.2 nM T84631 CYKJ28 44571092 IC50 = 5.4 nM T84631 CL9XM5 44571093 IC50 = 12 nM T84631 C0RU9L 44571134 IC50 = 1.8 nM T84631 C4BN3H 44573109 Ki = 10000 nM T84631 COR57Y 44573272 Ki = 4400 nM T84631 C6DX3Y 44573273 Ki = 3400 nM T84631 CM2R1P 44573274 Ki = 44000 nM T84631 CSP1I0 44573310 Ki = 2500 nM T84631 C6EG9V 44573311 Ki = 11000 nM T84631 CYV3X2 44573378 Ki = 17000 nM T84631 CWUA41 44573379 Ki = 100 nM T84631 CYA64G 44573380 Ki = 127000 nM T84631 CLG42S 44573428 Ki = 30000 nM T84631 C5F9RK 44577595 IC50 = 400 nM T84631 CIO19Z 44577596 IC50 = 1159 nM T84631 CLUJ07 44577597 IC50 = 246 nM T84631 CU2E3N 44577598 IC50 = 208 nM T84631 CC7IV5 44577599 IC50 = 494 nM T84631 C1LM4B 44577642 IC50 = 245 nM T84631 C5Q6ZB 44577643 IC50 = 276 nM T84631 CTE9W4 44577644 IC50 = 709 nM T84631 CD6OY9 44577645 IC50 = 193 nM T84631 C1O6VJ 44577646 IC50 = 227 nM T84631 CD2NO7 44577647 IC50 = 403 nM T84631 CX14HM 44577648 IC50 = 872 nM T84631 CV21YL 44577649 IC50 = 628 nM T84631 CO19SA 44577650 IC50 = 380 nM T84631 CVMN47 44577651 IC50 = 14 nM T84631 C3YZF4 44577954 IC50 = 517 nM T84631 CMK2S5 44577955 IC50 = 371 nM T84631 CP62MY 44577956 IC50 = 198 nM T84631 CRW83N 44577957 IC50 = 835 nM T84631 C01HVO 44577990 IC50 = 373 nM T84631 CPUZ06 44577991 IC50 = 222 nM T84631 C4XKY0 44577992 IC50 = 271 nM T84631 C30CBZ 44577993 IC50 = 396 nM T84631 CU4T1V 44577994 IC50 = 267 nM T84631 C15TZO 44577995 IC50 = 294 nM T84631 C65QDR 44577996 IC50 = 546 nM T84631 CF63WE 44578029 IC50 = 256 nM T84631 CHS79J 44578030 IC50 = 368 nM T84631 C5TBZ9 44578031 IC50 = 272 nM T84631 C3W8PT 44578032 IC50 = 462 nM T84631 CPYZ70 44578033 IC50 = 386 nM T84631 C7Y1QL 44578034 IC50 = 17 nM T84631 CLT8Z4 44578035 IC50 = 1073 nM T84631 CK6UG1 44578036 IC50 = 506 nM T84631 CLT5O2 44581199 Ki = 0.043 nM T84631 C97WFB 44581200 Ki = 0.084 nM T84631 CK8MJ1 44581201 Ki = 0.14 nM T84631 CPB78V 44581202 Ki = 0.74 nM T84631 CG1A0W 44581236 Ki = 0.56 nM T84631 C90ZBV 44581286 Ki = 0.18 nM T84631 CYL1B8 44581287 Ki = 0.32 nM T84631 CUJ83A 44581288 Ki = 0.071 nM T84631 CO12AM 44581325 Ki = 0.29 nM T84631 CHM16K 44581326 Ki = 0.59 nM T84631 C5CW2I 44581328 Ki = 0.36 nM T84631 C5BIF8 44581330 Ki = 0.068 nM T84631 CR75GK 44581361 Ki = 0.24 nM T84631 CH4M0F 44581362 Ki = 0.055 nM T84631 CB1GN5 44581363 Ki = 0.15 nM T84631 C2PXK1 44581390 Ki = 0.051 nM T84631 C6JX8N 44581393 Ki = 0.054 nM T84631 CT2DU0 44581418 Ki = 0.027 nM T84631 CMHW28 44581420 Ki = 0.042 nM T84631 CN32IF 44581421 Ki = 0.093 nM T84631 C8XF5J 44581456 Ki = 0.073 nM T84631 CA54PQ 44581457 Ki = 0.24 nM T84631 C2MQ1A 44581459 Ki = 0.11 nM T84631 CR42LZ 44581460 Ki = 0.78 nM T84631 CYZN78 44581494 Ki = 0.16 nM T84631 C2M3XU 44581496 Ki = 0.085 nM T84631 CLRP24 44581497 Ki = 0.12 nM T84631 C7ZQF0 44581498 Ki = 0.14 nM T84631 CMY6U3 44581556 Ki = 5.1 nM T84631 CN69DU 44581557 Ki = 3 nM T84631 CZ4L9O 44581558 Ki = 11 nM T84631 C7IKA3 44581559 Ki = 1.5 nM T84631 C9P7CT 44581590 Ki = 2.9 nM T84631 CBE98L 44581591 Ki = 7.6 nM T84631 C4N6LC 44581592 Ki = 20 nM T84631 CXW8T5 44581593 Ki = 0.55 nM T84631 C03LRJ 44581629 Ki = 0.02 nM T84631 CYUF13 44581630 Ki = 0.02 nM T84631 C6YDN5 44581631 Ki = 0.21 nM T84631 CJL04I 44581664 Ki = 0.021 nM T84631 C0UET1 44581665 Ki = 0.16 nM T84631 C6MTH1 44581704 Ki = 4.9 nM T84631 CX0T1R 44581705 Ki = 1.1 nM T84631 C6Y7QO 44581749 Ki = 0.065 nM T84631 CH6VU9 44581750 Ki = 0.31 nM T84631 C7Q8RG 44582128 IC50 = 0.5 nM T84631 CE4F0K 44582129 IC50 = 0.18 nM T84631 CN3FT7 44582147 IC50 = 1.2 nM T84631 C2LKP1 44582148 IC50 = 0.11 nM T84631 C4LZJ3 44582149 IC50 = 0.34 nM T84631 CA2N1I 44582150 IC50 = 0.02 nM T84631 CRW3K7 44582204 IC50 = 0.54 nM T84631 CIW63Z 44582205 IC50 = 0.31 nM T84631 C3E4LY 44582206 IC50 = 0.5 nM T84631 CCU71D 44582207 IC50 = 0.18 nM T84631 C0AG3O 44582221 IC50 = 0.22 nM T84631 CU5W8N 44582222 IC50 = 0.05 nM T84631 C06BKE 44582223 IC50 = 0.16 nM T84631 CJ96RG 44582224 IC50 = 0.08 nM T84631 C18TMJ 44586926 IC50 = 110 nM T84631 CR1XF9 44586927 IC50 = 840 nM T84631 C45DAE 44586955 IC50 = 75 nM T84631 C72KMC 44586956 IC50 = 88 nM T84631 CB8T1E 44586957 IC50 = 16 nM T84631 CCU92M 44586958 IC50 = 12 nM T84631 CR6X5Q 44587208 Ki = 2700 nM T84631 C87KXE 44587209 Ki = 330 nM T84631 CGOR19 44587231 Ki = 1500 nM T84631 C8WH9R 44587232 Ki = 160 nM T84631 C3WOP7 44587261 Ki = 25000 nM T84631 CX1DP6 44587262 Ki = 1800 nM T84631 C7K6JN 44587263 Ki = 3130 nM T84631 CKL1J2 44587264 Ki = 685 nM T84631 CTF79D 44587290 Ki = 2483 nM T84631 CBXY02 44587291 Ki = 14700 nM T84631 CDBV80 44587292 Ki = 5700 nM T84631 CWZ34J 44587314 Ki = 920 nM T84631 C6Y1FA 44587835 Ki = 3000 nM T84631 C91QNS 44587836 Ki = 14000 nM T84631 C0CRG4 44589267 IC50 = 336 nM T84631 CY3VQ2 44589268 IC50 = 46 nM T84631 C10NMD 44590397 Ki = 7991 nM T84631 COQ0E6 44592399 IC50 = 35 nM T84631 CK82XN 44592400 IC50 = 290 nM T84631 C3XEW7 44592401 IC50 = 25 nM T84631 C96CWM 44592402 IC50 = 30 nM T84631 C17NRH 44592470 IC50 = 6 nM T84631 CRF34H 44592525 IC50 = 9 nM T84631 C3L1AN 44592526 IC50 = 8 nM T84631 CI5C1F 44592560 IC50 = 26.96 nM T84631 C9RWU8 44592561 IC50 = 0.31 nM T84631 CHK9G2 44592562 IC50 = 6.62 nM T84631 CNIX06 44592593 IC50 = 11.27 nM T84631 CZJ7C6 44592617 IC50 = 46.05 nM T84631 C1A8YB 44592658 IC50 = 50 nM T84631 CN7G0O 44592693 IC50 = 36.49 nM T84631 CC65UK 44592729 IC50 = 1.3 nM T84631 C9OG6N 44592765 IC50 = 0.05 nM T84631 CKC2Q8 44592831 IC50 = 0.13 nM T84631 CY2IM4 44592833 IC50 = 0.05 nM T84631 CW72YN 44592864 IC50 = 0.02 nM T84631 CD4G2B 44592865 IC50 = 0.23 nM T84631 CDLY78 44592888 IC50 = 1.75 nM T84631 C4RDW0 44592955 IC50 = 50 nM T84631 C1PLT5 44592978 IC50 = 50 nM T84631 CVS21G 44592979 IC50 = 8.14 nM T84631 C4M0KI 44593006 IC50 = 1.17 nM T84631 C9PCO6 44593008 IC50 = 7.6 nM T84631 C1Y8IM 44593413 Ki = 0.064 nM T84631 C8X3KA 44593414 Ki = 0.025 nM T84631 C97UBM 44593556 IC50 = 7.5 nM T84631 CPZR42 44607103 IC50 = 27900 nM T84631 C6MIK9 44626665 IC50 = 1023 nM T84631 C4LQW3 44629430 Ki = 11900 nM T84631 CL20GE 44629584 Ki = 0.2 nM T84631 CUK2I7 45103480 Ki = 70 nM T84631 CP6SB1 45103481 Ki = 290 nM T84631 CM16YW 45103482 Ki = 52 nM T84631 C2PVE0 45103523 Ki = 6500 nM T84631 CKN2F4 45103582 Ki = 2.6 nM T84631 C80DXA 45103583 Ki = 0.5 nM T84631 CG51EA 45103584 Ki = 1300 nM T84631 C46JPW 45103585 Ki = 250 nM T84631 C8XBZ6 45103586 Ki = 560 nM T84631 CXS6K8 45103587 Ki = 825 nM T84631 CPR1O7 45103680 Ki = 354 nM T84631 CJU8M5 45103681 Ki = 2844 nM T84631 CZ4JW1 45261445 Ki = 102 nM T84631 C3P8EA 45263195 IC50 = 600 nM T84631 CK7E3M 45264760 Ki = 220 nM T84631 C3Y8WE 45266133 Ki = 3900 nM T84631 C5E6AS 45267012 IC50 = 1720 nM T84631 CZ32WR 45267285 IC50 = 2882 nM T84631 C1TYA3 45267286 IC50 = 2677 nM T84631 CU3WJ8 45267299 IC50 = 21 nM T84631 C41ELS 45267302 IC50 = 928 nM T84631 C67DKE 45267303 IC50 = 195 nM T84631 CGU67A 45267836 IC50 = 2030 nM T84631 CW3SX0 45267838 IC50 = 1050 nM T84631 CT1WY2 45268147 IC50 = 780 nM T84631 C1ZWU3 45268157 IC50 = 2600 nM T84631 CCVL15 45268158 IC50 = 2939 nM T84631 CB1O0D 45268159 IC50 = 11 nM T84631 C6GDW5 45268170 IC50 = 53 nM T84631 CY75OX 45268711 IC50 = 2810 nM T84631 CZ0YE8 45269033 IC50 = 11879 nM T84631 CMSU50 45269045 IC50 = 30000 nM T84631 C9Z5TG 45269048 IC50 = 15 nM T84631 CSY60N 45269572 IC50 = 3230 nM T84631 CO18RA 45269846 IC50 = 54 nM T84631 C42QBM 45269847 IC50 = 28 nM T84631 C2QLJ7 45269887 IC50 = 2400 nM T84631 CDAM80 45269891 IC50 = 349 nM T84631 CQO6T8 45269898 IC50 > 32000 nM T84631 COA86N 45270402 IC50 = 1520 nM T84631 CFQ14D 45270405 IC50 = 800 nM T84631 CH1P5M 45270407 IC50 = 2790 nM T84631 CP7DF5 45270707 IC50 > 34000 nM T84631 C7EV9T 45270708 IC50 > 34000 nM T84631 CAMB38 45270720 IC50 = 76 nM T84631 CI49ER 45270731 IC50 = 19 nM T84631 C90JGW 45270732 IC50 = 386 nM T84631 CB2QX3 45270733 IC50 = 22 nM T84631 C6YPG9 45270763 Ki = 14 nM T84631 CU26GQ 45271227 IC50 = 1630 nM T84631 C41TXV 45271542 IC50 = 167 nM T84631 C45DVC 45271581 Ki = 43 nM T84631 CW6CB5 45272126 IC50 = 210 nM T84631 CWP6T9 45272400 IC50 = 5 nM T84631 CPBF26 45272436 IC50 > 34000 nM T84631 C96EXW 45272443 IC50 = 18759 nM T84631 C49XBD 45272455 IC50 = 940 nM T84631 C7UDO4 45273309 IC50 = 1300 nM T84631 CF97AM 45273310 IC50 = 84 nM T84631 C4N0LV 45273311 IC50 = 15538 nM T84631 C69XFH 45273319 IC50 = 2728 nM T84631 CS8U0D 45273320 IC50 = 27 nM T84631 CQ7SY8 45273327 IC50 = 14818 nM T84631 CJ73BT 45486346 Ki = 83000 nM T84631 C9ETC4 45486354 Ki = 123000 nM T84631 CVEK34 45488045 IC50 = 18 nM T84631 CK15WB 45488046 IC50 = 10 nM T84631 CE4F6R 45488047 IC50 = 3 nM T84631 CI5S4V 45488048 IC50 = 3 nM T84631 C8VOL9 46191308 Ki = 0.8 nM T84631 CCG5U1 46196561 Ki = 0.5 nM T84631 C1I0OD 46222444 IC50 = 11 nM T84631 CCP8B0 46222445 IC50 = 1.7 nM T84631 CCM09Y 46222669 IC50 = 24 nM T84631 CCH8I6 46222670 IC50 = 51 nM T84631 CQ4BV0 46222671 IC50 = 60 nM T84631 C14DQZ 46222672 IC50 = 14 nM T84631 C9LU7N 46222673 IC50 = 147 nM T84631 C5T6FE 46226298 Ki = 6.2 nM T84631 CB9O0A 46226299 Ki = 6 nM T84631 CW86BU 46226322 Ki = 5.1 nM T84631 CV1R9H 46226323 Ki = 35 nM T84631 C8JPB3 46226324 Ki = 1.5 nM T84631 C63LKZ 46226325 Ki = 0.8 nM T84631 C3WRU1 46226349 Ki = 5 nM T84631 CS7X8I 46226372 Ki = 0.8 nM T84631 C3IA0F 46226373 Ki = 2 nM T84631 CE6F8R 46226374 Ki = 1 nM T84631 C1HPB8 46226391 Ki = 5 nM T84631 CGZF19 46226392 Ki = 0.8 nM T84631 CO8I9D 46226393 Ki = 2 nM T84631 CG8LX3 46226394 Ki = 2 nM T84631 CKL39P 46226415 Ki = 4 nM T84631 CQW85G 46226416 Ki = 2 nM T84631 C3RMI8 46226796 IC50 > 5000 nM T84631 C7BQ1U 46226806 IC50 = 21 nM T84631 CM10IF 46226817 IC50 = 930 nM T84631 CW47XK 46232635 Ki = 9 nM T84631 C9L1ZS 46233075 Ki = 1560 nM T84631 CD62VO 46233076 Ki = 1270 nM T84631 C5PI6E 46233077 Ki = 1300 nM T84631 C9BLH7 46233114 Ki = 2375 nM T84631 C42DOH 46233115 Ki = 1628 nM T84631 CA7S2F 46233116 Ki = 1585 nM T84631 CQ4UF5 46233117 Ki = 2115 nM T84631 CEU41B 46233150 Ki = 1363 nM T84631 CXV4P6 46233151 Ki = 3970 nM T84631 CFA7H0 46233153 Ki = 2600 nM T84631 CH01MJ 46233194 Ki = 600 nM T84631 CR5VN4 46233261 Ki = 6200 nM T84631 CHF74W 46233262 Ki = 7300 nM T84631 C8ONP6 46233306 Ki = 4300 nM T84631 CG6QI5 46233307 Ki = 2900 nM T84631 CL0W5E 46233309 Ki = 4300 nM T84631 C8AQZ5 46233310 Ki = 13100 nM T84631 C7XT0F 46233339 Ki = 7900 nM T84631 CJ3P5N 46233341 Ki = 5700 nM T84631 CBC4Y5 46233342 Ki = 105 nM T84631 CUPC52 46233343 Ki = 55 nM T84631 CHF45Z 46233364 Ki > 100000 nM T84631 CUZW20 46233366 Ki = 3350 nM T84631 CTMN13 46233367 Ki = 1150 nM T84631 C23KIW 46233369 Ki = 45000 nM T84631 CLHX82 46233406 Ki = 13800 nM T84631 C8T5CW 46233408 Ki = 3400 nM T84631 CQ01MF 46233409 Ki = 150 nM T84631 CY92TG 46233410 Ki = 950 nM T84631 CZ7CQ8 46233411 Ki = 44 nM T84631 CPBS35 46233412 Ki = 910 nM T84631 C12SEZ 46233413 Ki = 17 nM T84631 C7VKZ8 46233414 Ki = 33 nM T84631 CCI75A 46233462 Ki = 37 nM T84631 CYG6A2 46233463 Ki = 25 nM T84631 CT5MH6 46233491 Ki = 0.6 nM T84631 CY5C1O 46233492 Ki = 4450 nM T84631 C5H2EF 46233511 Ki = 960 nM T84631 CZ46CU 46233512 Ki = 1740 nM T84631 CI8NV4 46233513 Ki = 700 nM T84631 C84HTG 46233514 Ki = 360 nM T84631 CA4Z5X 46233537 Ki = 1810 nM T84631 C5SK7C 46233538 Ki = 830 nM T84631 C0Y8IT 46233539 Ki = 550 nM T84631 C16IMD 46233540 Ki = 1300 nM T84631 CW3S0U 46233565 Ki = 1700 nM T84631 C03TRU 46233566 Ki = 1184 nM T84631 C8RCY2 46233567 Ki = 800 nM T84631 CHO28I 46233568 Ki = 600 nM T84631 CRDC20 46233603 Ki = 3773 nM T84631 CWVY84 46233604 Ki = 872 nM T84631 C7ZP4M 46233605 Ki = 1562 nM T84631 CT84CW 46233649 Ki = 1147 nM T84631 CF8Z3Q 46233651 Ki = 828 nM T84631 CX28UI 46233688 Ki = 1482 nM T84631 C9P0FC 46233689 Ki = 1303 nM T84631 CWO0V7 46233690 Ki = 2252 nM T84631 C7ET8Q 46233691 Ki = 2051 nM T84631 C8E0ZQ 46835134 Ki = 192 nM T84631 C62RBC 46835135 Ki = 9 nM T84631 CY47OV 46878192 Ki > 6000 nM T84631 CQ2G6A 46878194 Ki > 6000 nM T84631 CC6GE9 46878197 Ki = 970 nM T84631 CE79OB 46878198 Ki > 6000 nM T84631 CS07EW 46878199 Ki > 6000 nM T84631 C3HZP7 46878200 Ki = 6000 nM T84631 CF5ZQ8 46878201 Ki = 6000 nM T84631 C7ICJ0 46878202 Ki > 6000 nM T84631 CQJR51 46878203 Ki = 9 nM T84631 C9BXU7 46878204 Ki = 6000 nM T84631 CXQL63 46878205 Ki > 6000 nM T84631 CR93NC 46878206 Ki > 6000 nM T84631 C0H3UO 46878241 Ki > 5000 nM T84631 CS7B4G 46888797 IC50 = 20 nM T84631 CNS8R6 46888834 IC50 = 49 nM T84631 CPT7U3 46888835 IC50 = 28 nM T84631 CS7XO5 46889240 IC50 = 23 nM T84631 C9E3HU 46889265 IC50 = 46 nM T84631 C8U3OW 46889266 IC50 = 198 nM T84631 CNA06P 46905365 Ki = 200 nM T84631 CX2L8G 46905375 Ki = 34 nM T84631 CTR32W 46905376 Ki = 10 nM T84631 CS8GZ7 46905377 Ki = 200 nM T84631 C9W1ZK 46905378 Ki = 670 nM T84631 CR6P1E 46905379 Ki = 71 nM T84631 C75IRP 46905995 Ki = 1.3 nM T84631 CB2F7T 46978227 Ki > 62500 nM T84631 CEDL20 49796469 Ki = 80 nM T84631 C8NK1S 49796470 Ki = 800 nM T84631 C4MK5H 49796471 Ki = 7800 nM T84631 C75HOB 49796472 Ki = 900 nM T84631 CS90ZF 49796473 Ki = 24 nM T84631 CXUM36 49820499 Ki = 300 nM T84631 CX7SA8 49820500 Ki = 300 nM T84631 C6OIW8 49820657 Ki = 2300 nM T84631 CAI5S9 49827569 Ki = 7.943 nM T84631 CU1DK9 49835415 Ki = 52 nM T84631 C0OQ8N 49835557 Ki = 2.7 nM T84631 CQ23SL 49864307 Ki = 201 nM T84631 CTO73I 49864308 Ki = 22 nM T84631 CT8NM4 49864309 Ki = 46 nM T84631 C8U1HB 49864310 Ki = 40 nM T84631 C78QKE 49864328 Ki = 120 nM T84631 CFIW73 49864329 Ki = 28 nM T84631 CDZ3B0 49864350 Ki = 11 nM T84631 CLW9I6 49864373 Ki = 17 nM T84631 CSZ3P1 49864435 Ki = 46 nM T84631 CZR1W9 49864436 Ki = 34 nM T84631 C5YH3T 49864437 Ki = 44 nM T84631 CK5G4W 49864458 Ki = 11 nM T84631 CLOY62 49864459 Ki = 24 nM T84631 CR8JK9 49864483 Ki = 27 nM T84631 C42KOC 49864498 Ki = 345 nM T84631 CR3F4Q 49864657 Ki = 36 nM T84631 CIP8O4 49864658 Ki = 92 nM T84631 CWA50O 49864685 Ki = 1779 nM T84631 C9P6TE 49864704 Ki = 42 nM T84631 CM4YA0 49864705 Ki = 15 nM T84631 CRW92J 49864706 Ki = 40 nM T84631 CU0LX7 50919254 Ki = 2 nM T84631 C2LK1E 50919255 Ki = 9 nM T84631 CIZ5Y1 50919256 Ki = 2 nM T84631 CC89AZ 50919257 Ki = 4 nM T84631 CAM3V7 50939649 Ki = 50 nM T84631 CHC74O 50939651 Ki = 810 nM T84631 CT9P8Q 51041296 Ki = 0.11 nM T84631 CKCN49 51346898 Ki = 3 nM T84631 CV0IQ5 52940898 Ki < 0.3 nM T84631 C2DO1B 52940908 IC50 = 8 nM T84631 C84CYB 52940909 IC50 = 4 nM T84631 C4FDU5 52941018 IC50 = 35 nM T84631 C1DRJ2 52941698 Ki = 0.1 nM T84631 C57MVG 52942150 Ki = 3 nM T84631 CPK9R0 52943286 Ki = 0.7 nM T84631 CBO9N7 52943447 IC50 = 120 nM T84631 CQ19NI 52944468 Ki = 2 nM T84631 C1M3EC 52944526 IC50 = 3 nM T84631 C1RWG9 52944684 IC50 = 3450 nM T84631 C8XN9J 52945796 Ki = 1100 nM T84631 CR06QB 52946959 Ki = 0.55 nM T84631 CI0P3R 52947731 Ki = 0.9 nM T84631 CU90GX 52949410 Ki < 0.4 nM T84631 CVRQ75 52949419 Ki = 0.6 nM T84631 C4Y8FZ 52949515 Ki = 16000 nM T84631 CPE05T 53242224 IC50 = 2.2 nM T84631 CB8XU4 53317105 IC50 = 13 nM T84631 CS6TR3 53317106 IC50 = 48 nM T84631 COP4X3 53317127 IC50 = 9 nM T84631 CX1KR9 53317330 Ki = 1 nM T84631 CA86OS 53317375 Ki = 1000000 nM T84631 CA45BG 53317639 IC50 = 1618 nM T84631 C8U3NB 53317693 IC50 = 439 nM T84631 C68TOQ 53318416 IC50 = 1930 nM T84631 CIVY68 53318619 Ki = 15 nM T84631 CXVJ49 53318620 Ki = 6 nM T84631 CLUD64 53319727 IC50 = 4145 nM T84631 CWOK94 53321019 IC50 = 27 nM T84631 C6K1WJ 53321020 IC50 = 11 nM T84631 C79RGN 53321237 Ki = 5 nM T84631 CAYD14 53321238 Ki = 2 nM T84631 C7QEI1 53321291 Ki = 16000 nM T84631 C7CR5Q 53322361 IC50 = 6830 nM T84631 CL0SC2 53322387 IC50 = 623 nM T84631 CL6R7Y 53322388 IC50 = 204 nM T84631 CL29IO 53322566 Ki = 6 nM T84631 CFOI53 53322612 Ki = 80000 nM T84631 CR0VJ3 53323722 IC50 = 93 nM T84631 C3B1AG 53323723 IC50 = 2476 nM T84631 C0A1DL 53323905 Ki = 2 nM T84631 CWA7B3 53323948 Ki = 1000000 nM T84631 CUQ82T 53324997 IC50 = 1025 nM T84631 CJB75L 53324998 IC50 = 5675 nM T84631 CP9JT3 53324999 IC50 = 18 nM T84631 CSHU35 53325000 IC50 = 12 nM T84631 CO6TG4 53325236 Ki = 1000000 nM T84631 CO0R2M 53325237 Ki = 1000000 nM T84631 COF8N6 53325369 Ki = 3 nM T84631 CK25QS 53326291 IC50 = 642 nM T84631 CFB65G 53326292 IC50 > 10000 nM T84631 CW10IE 53326477 Ki = 100 nM T84631 CT2RQ6 53326832 Ki = 4 nM T84631 C0DYJ6 53326870 IC50 = 59 nM T84631 CA6GQ5 53341037 Ki > 13300 nM T84631 CIKQ81 53345652 Ki > 130 nM T84631 CXWS90 53345968 Ki > 1000 nM T84631 CB08CW 53379392 Ki = 129 nM T84631 C6XNM0 53380822 Ki = 1500 nM T84631 C1KFQ0 53380823 Ki = 9800 nM T84631 C7JWD0 53380936 Ki = 6660 nM T84631 C97KGD 53380937 Ki = 6800 nM T84631 CKV6Q2 53380938 Ki = 1600 nM T84631 C47WIH 53380939 Ki = 15000 nM T84631 CY3RO0 53380940 Ki = 5490 nM T84631 C3R8PW 53380941 Ki = 6000 nM T84631 CI5XO8 53388478 IC50 = 970000 nM T84631 C4HB3V 53392251 IC50 > 300000 nM T84631 CV60BK 53488415 Ki = 4.71 nM T84631 C8SCH2 53800364 IC50 = 50 nM T84631 C9GFU3 53864431 IC50 = 190 nM T84631 C16KAQ 53954748 IC50 = 56 nM T84631 CEIQ26 54352954 IC50 = 3000 nM T84631 CQNW76 54507330 IC50 = 200 nM T84631 C2FS3H 54555233 IC50 = 100 nM T84631 CI67SD 54580287 IC50 = 1600 nM T84631 C82FQT 54580288 IC50 = 3.5 nM T84631 C4C3DP 54581293 IC50 = 200 nM T84631 CXE31M 54581294 IC50 = 7.4 nM T84631 CV20EN 54581295 IC50 > 10000 nM T84631 CUY6J3 54581296 IC50 = 65 nM T84631 CE3D7F 54582336 IC50 = 1.9 nM T84631 C3EM0S 54583288 IC50 = 3945 nM T84631 CUSC68 54583289 IC50 = 7.7 nM T84631 C9IJ0M 54583290 IC50 = 170 nM T84631 C6C7NO 54584026 Ki = 0.5012 nM T84631 CH3A5X 54584246 IC50 = 1200 nM T84631 CYB6H9 54584247 IC50 = 970 nM T84631 C2H6IJ 54584248 IC50 = 110 nM T84631 C0MA2W 54584249 IC50 = 1.1 nM T84631 CSMJ20 54584250 IC50 = 2.5 nM T84631 C38YZE 54584279 IC50 = 120 nM T84631 CN7T4Q 54584280 IC50 = 100 nM T84631 CC1S7R 54585216 IC50 = 70 nM T84631 C7TEM9 54585217 IC50 = 770 nM T84631 CL86NU 54585218 IC50 = 5.6 nM T84631 CP8EA5 54585238 IC50 = 2.7 nM T84631 C7BTJ1 54586167 IC50 = 47 nM T84631 CC6AT1 54586168 IC50 = 460 nM T84631 CT8G6K 54586169 IC50 = 610 nM T84631 C5K3JQ 54586170 IC50 = 100 nM T84631 CBO8V7 54587183 IC50 = 221 nM T84631 CNO24S 54587184 IC50 = 4100 nM T84631 CQ5PV6 54587185 IC50 = 2100 nM T84631 CFLR93 54587186 IC50 = 29 nM T84631 C2GZA5 54587362 IC50 = 690 nM T84631 C9I4OP 54738720 Ki = 4400 nM T84631 CWQ17K 54751669 Ki = 146 nM T84631 CK52NT 54751670 Ki = 1620 nM T84631 C17MSO 56640092 Ki = 152 nM T84631 CGP7Y6 56640160 Ki = 21 nM T84631 C30AJK 56640226 Ki = 784 nM T84631 C9YXM2 56659587 IC50 = 1078000 nM T84631 CA32CM 56659850 Ki = 1.4 nM T84631 C6OI5V 56660094 Ki = 8000 nM T84631 CKFI81 56660095 Ki = 1200 nM T84631 CKO4M6 56663319 Ki = 37 nM T84631 C2T1WM 56665604 IC50 = 380 nM T84631 CMG9H6 56666511 IC50 > 580000 nM T84631 CCM80T 56670171 Ki = 31 nM T84631 C0M3AE 56673432 IC50 > 1480000 nM T84631 CI6RX7 56673433 IC50 > 590000 nM T84631 CGM2J4 56673694 Ki = 21 nM T84631 C4T6NO 56673695 Ki = 14.5 nM T84631 C7DE8I 56676739 IC50 > 1340000 nM T84631 CE4AT6 56676740 IC50 > 400000 nM T84631 C8CN9W 56676741 IC50 = 440000 nM T84631 C1TH3W 56677006 Ki = 565 nM T84631 CY34VE 56677007 Ki = 2.1 nM T84631 C5LVJ2 56680051 IC50 > 640000 nM T84631 CKF2M0 56680052 IC50 = 508000 nM T84631 C72IHP 56680339 Ki = 397 nM T84631 CT7U8L 56683905 Ki = 4900 nM T84631 C3CDB4 56683906 Ki = 4700 nM T84631 C14YLP 56849975 IC50 = 103 nM T84631 C5DQ2M 56849977 IC50 = 539 nM T84631 C1F8IX 56849978 IC50 = 140 nM T84631 C2V0JC 56850120 IC50 = 73.4 nM T84631 CRL87T 56850121 IC50 = 118 nM T84631 CKD9E0 56850122 IC50 = 213 nM T84631 CIDT59 56850256 IC50 = 99.2 nM T84631 CE0X3B 56850258 IC50 = 31.1 nM T84631 CFZ7P2 56850260 IC50 = 50.3 nM T84631 C06NPR 56850396 IC50 = 157 nM T84631 CN35WB 56850397 IC50 = 155 nM T84631 CLS9Y7 56850526 IC50 = 1438 nM T84631 CKNE35 56850528 IC50 = 6143 nM T84631 CX63IV 56850529 IC50 = 349 nM T84631 CN5EI8 56850671 IC50 = 64.2 nM T84631 CM2W4G 56850672 IC50 = 59.8 nM T84631 CJAK41 56850673 IC50 = 86.1 nM T84631 CDKY37 56850674 IC50 = 41.3 nM T84631 CLF6Q0 56850675 IC50 = 41.4 nM T84631 C8UHN3 56949979 IC50 = 9000 nM T84631 CH1EI8 56954620 Ki = 3430 nM T84631 C4EHU8 56954732 Ki = 9370 nM T84631 C5C8XO 56954733 Ki = 3472 nM T84631 CST4F0 56954834 Ki = 42 nM T84631 CRK92A 56954952 Ki = 1860 nM T84631 CB57DW 57391171 Ki = 7600 nM T84631 CZ6D2Q 57391429 IC50 = 4.9 nM T84631 CZ41MI 57391430 IC50 = 0.74 nM T84631 CWJ4I7 57391565 Ki = 14000 nM T84631 C36LXQ 57392276 IC50 = 20 nM T84631 CPBW48 57392333 Ki = 360000 nM T84631 CUI1W3 57392347 IC50 = 32 nM T84631 CPF25Q 57392348 IC50 = 337 nM T84631 C15EGS 57392349 IC50 = 674 nM T84631 C0DZ6H 57392472 IC50 = 7 nM T84631 C7APO2 57392934 Ki = 6500 nM T84631 CZ2A0S 57392935 Ki = 1600 nM T84631 C6M5RS 57393195 IC50 = 1.6 nM T84631 CX16KB 57393324 Ki = 4000 nM T84631 CG9AS5 57394027 IC50 = 8.3 nM T84631 C1AZB4 57394031 IC50 = 4.7 nM T84631 CR9S5P 57394086 IC50 = 129 nM T84631 CNQT87 57394087 IC50 = 1330 nM T84631 COB56U 57394088 IC50 = 22 nM T84631 C3K0VW 57394177 IC50 = 13 nM T84631 C6EWL9 57394677 Ki = 5600 nM T84631 CE2BA9 57394917 IC50 = 49 nM T84631 CG07ZY 57394918 IC50 = 1.5 nM T84631 C8T2ZJ 57395044 Ki = 790 nM T84631 CNLD49 57395793 IC50 = 5 nM T84631 CL2JE5 57395841 Ki = 310000 nM T84631 CSF3D7 57395856 IC50 = 32 nM T84631 CN0UR9 57395857 IC50 = 51 nM T84631 CI1QX2 57395858 IC50 = 14 nM T84631 C2JI3K 57397571 IC50 = 6 nM T84631 CKR94L 57397646 IC50 = 11 nM T84631 CYEK40 57397750 IC50 = 10 nM T84631 C9F4OL 57398232 Ki = 7700 nM T84631 C5OAB7 57398233 Ki = 2830 nM T84631 CY39KP 57398234 Ki = 1600 nM T84631 C83YUW 57398444 IC50 = 53 nM T84631 C9MWA3 57399250 IC50 = 4.8 nM T84631 C49TVR 57399313 IC50 = 121 nM T84631 C7F4ER 57399314 IC50 = 1957 nM T84631 CRQ19W 57399315 IC50 = 209 nM T84631 C5SK3Q 57399481 IC50 = 1110 nM T84631 CODX48 57399879 Ki = 18000 nM T84631 C93VSX 57399880 Ki = 4100 nM T84631 C5WOZ3 57399881 Ki = 3600 nM T84631 CC69OL 57400113 IC50 = 9.1 nM T84631 CUX76O 57400114 IC50 = 2.4 nM T84631 C9ZL5X 57400230 Ki = 1600 nM T84631 CPZR79 57400272 Ki = 6600 nM T84631 CKYJ43 57401018 IC50 = 6.3 nM T84631 CH2AN8 57401242 IC50 = 9750 nM T84631 CS2ZY1 57401658 Ki = 16300 nM T84631 C92EDA 57401914 IC50 = 231 nM T84631 C7F3ET 57401915 IC50 = 4.9 nM T84631 C7SM8P 57401916 IC50 = 2.9 nM T84631 CJ9TH7 57402084 IC50 = 1.2 nM T84631 CH90JO 57402841 IC50 = 130 nM T84631 C6T0ZQ 57402842 IC50 = 14 nM T84631 C0H4UQ 57402934 IC50 = 32 nM T84631 CG90KP 57403382 Ki = 7700 nM T84631 C3CKA6 57403383 Ki = 4400 nM T84631 C4OB6Z 57403384 Ki = 14000 nM T84631 CD0XJ5 57403637 IC50 = 6.9 nM T84631 CDW0N6 57403638 IC50 = 2 nM T84631 CKI4S8 57403776 Ki = 9800 nM T84631 C5MX2D 57404340 IC50 > 50000 nM T84631 C4R2LU 57594784 IC50 = 4.9 nM T84631 C5NC8T 57594789 IC50 = 15 nM T84631 C63FQC 57803696 Ki = 460 nM T84631 CLV91D 57803729 Ki = 4070 nM T84631 CEH39Z 57803776 Ki = 2330 nM T84631 C2W7GY 57803799 Ki = 560 nM T84631 CU4N3X 57803861 Ki = 680 nM T84631 CEG27C 57803875 Ki = 450 nM T84631 CI6U8B 57803906 Ki = 760 nM T84631 C6X3ER 57803948 Ki = 540 nM T84631 CH2QT8 57804013 Ki = 430 nM T84631 C45OXB 57804023 Ki = 2190 nM T84631 CFMO72 57804069 Ki = 430 nM T84631 CTE30K 57842560 Ki = 4800 nM T84631 C0C6UB 57842624 Ki = 3300 nM T84631 C7XY5A 57842673 Ki > 9000 nM T84631 CU9S6K 57842710 Ki = 2600 nM T84631 CL8T7M 57842742 Ki = 610 nM T84631 C41NSR 57842812 Ki = 5500 nM T84631 C9XW1C 57842830 Ki = 5800 nM T84631 CWF0C3 57842850 Ki = 3200 nM T84631 C73CPB 57842913 Ki = 1000 nM T84631 CB5F0H 57942680 Ki = 4500 nM T84631 C8GXF1 57942687 Ki = 6000 nM T84631 CO52PA 57942693 Ki = 6400 nM T84631 CS23DW 57942743 Ki = 5200 nM T84631 C0DO5P 57942817 Ki = 5200 nM T84631 CV0KZ6 57942834 Ki = 3700 nM T84631 C0KRC1 57942835 Ki = 2900 nM T84631 C60HCV 57976401 Ki > 13300 nM T84631 CHB27Y 57976410 Ki = 1128 nM T84631 CM8UJ7 57976444 Ki > 1000 nM T84631 CQ71KE 57976446 Ki = 1500 nM T84631 CXL75F 58630486 Ki > 15000 nM T84631 C3OA5C 58789089 Ki = 3500 nM T84631 C2W1UT 58789135 Ki = 2800 nM T84631 CT9C1Z 58789193 Ki = 8200 nM T84631 C1C8SA 59019689 Ki = 1.5 nM T84631 CP2WM6 59019709 Ki = 0.15 nM T84631 CCM38Z 59020027 Ki = 0.2 nM T84631 C4R9VT 59020061 Ki = 0.05 nM T84631 C7NUC3 59020071 Ki = 1.22 nM T84631 C5ICF9 59020139 Ki = 0.06 nM T84631 CL6EP7 59020154 Ki = 0.48 nM T84631 CSC0L5 59020200 Ki = 0.66 nM T84631 C56MGU 59020231 Ki = 0.05 nM T84631 CDMI79 59020246 Ki = 0.07 nM T84631 CYF20E 59020269 Ki = 9.27 nM T84631 C91APY 59095797 IC50 = 270 nM T84631 C69SED 59095888 IC50 = 1700 nM T84631 CN09MI 59108388 IC50 = 68 nM T84631 C1BHM8 59108407 IC50 = 6.9 nM T84631 CPW2H7 59315536 Ki = 2800 nM T84631 CO38AC 59402011 Ki > 9000 nM T84631 CMU38J 59432238 IC50 = 1.5 nM T84631 CA83BF 59432241 IC50 = 66 nM T84631 C7IO5P 60150643 Ki = 900 nM T84631 C6JP8Q 60154989 Ki = 340 nM T84631 CE5A7B 60162406 Ki > 10000 nM T84631 C8TWY6 66554641 Ki = 6900 nM T84631 CUWT16 66554643 Ki = 0.25 nM T84631 C1W8HF 66554816 Ki = 0.09 nM T84631 CA8L6M 66573468 IC50 = 19000 nM T84631 C2CX0G 66573469 IC50 = 221000 nM T84631 C71CLE 66573471 IC50 = 12800 nM T84631 C8R7DY 66573472 IC50 = 19000 nM T84631 CG0O8A 66573532 IC50 = 20000 nM T84631 CP6JT5 66573533 IC50 = 6000 nM T84631 C6C3MI 66573535 IC50 = 42000 nM T84631 C9N5SP 66573536 IC50 = 56000 nM T84631 C5XP9E 66573589 IC50 = 209000 nM T84631 C8V9FN 66573590 IC50 = 19000 nM T84631 CP30LR 66573591 IC50 = 1300 nM T84631 CWT42D 66573592 IC50 = 14000 nM T84631 CJMT47 66573593 IC50 = 34000 nM T84631 CIR14C 66573637 IC50 = 197000 nM T84631 C2ELC3 66573638 IC50 = 85000 nM T84631 C1XS3L 66573639 IC50 = 335000 nM T84631 CQT4K0 66573640 IC50 = 246000 nM T84631 CTVP01 66573641 IC50 = 18000 nM T84631 C5JOZ8 66573709 IC50 = 900 nM T84631 CEJ02R 66573710 IC50 = 311000 nM T84631 CD86QN 66573711 IC50 = 13300 nM T84631 C2H9VX 66573712 IC50 = 103000 nM T84631 C8VZC9 66573779 IC50 = 1300 nM T84631 CM0DX8 66573780 IC50 = 36000 nM T84631 CKJG43 66573781 IC50 = 1100 nM T84631 CKY92Q 66573782 IC50 = 5400 nM T84631 C27HBF 66573783 IC50 = 190000 nM T84631 CA61DQ 66573843 IC50 > 500000 nM T84631 CZ6N3E 66573844 IC50 = 1600 nM T84631 CWCA65 66573845 IC50 = 270 nM T84631 C8MNG4 66573846 IC50 > 500000 nM T84631 CDL02G 66573847 IC50 = 2900 nM T84631 CH6VF3 66573909 IC50 > 500000 nM T84631 C5N8TC 66573910 IC50 = 151000 nM T84631 CXZ02D 66573911 IC50 > 500000 nM T84631 CY17TB 66573912 IC50 > 500000 nM T84631 CL9B6F 66573973 IC50 = 7800 nM T84631 CT4CR3 66573974 IC50 = 54000 nM T84631 CJG14M 66574033 IC50 > 500000 nM T84631 CR5IJ8 66574034 IC50 = 69000 nM T84631 CPV28L 66574037 IC50 = 371000 nM T84631 C3PV1H 66574099 IC50 = 358000 nM T84631 C5RZE9 66574100 IC50 = 99000 nM T84631 CNG0E4 66574102 IC50 = 23000 nM T84631 CFR0J7 66574158 IC50 = 9000 nM T84631 CBE3G1 66574160 IC50 = 10000 nM T84631 CS1B2I 66574390 IC50 = 9900 nM T84631 C09HIT 66574391 IC50 = 16400 nM T84631 C3LT2W 66674079 Ki > 8180 nM T84631 C23QOJ 66674821 Ki > 8180 nM T84631 CWOD93 66744646 Ki > 13300 nM T84631 CSAQ19 66818162 Ki = 400 nM T84631 C89BXR 66818555 Ki = 300 nM T84631 C9LTK3 66818589 Ki = 600 nM T84631 C41RKZ 66818743 Ki = 1500 nM T84631 CRH5O7 66818889 Ki = 200 nM T84631 CE6JP2 66911194 IC50 = 2.6 nM T84631 CGH09I 66911211 IC50 = 3.4 nM T84631 CKWQ82 67155200 Ki = 1 nM T84631 CY05ND 67155277 IC50 = 145 nM T84631 CA0GE1 67155403 IC50 = 1.1 nM T84631 CN51PD 67155431 IC50 = 1 nM T84631 C0SDB3 68020667 Ki = 7357 nM T84631 C17JAZ 68284084 IC50 > 30000 nM T84631 CE79VS 68440006 Ki = 5400 nM T84631 CA5DG8 69249482 Ki = 1300 nM T84631 CQY32W 69295008 Ki = 7300 nM T84631 CFPM31 69442778 IC50 = 150 nM T84631 C3BFL4 69515911 Ki = 0.07 nM T84631 CL5MN1 69516774 Ki = 0.24 nM T84631 CO7TI8 69516837 Ki = 1.01 nM T84631 CX10QE 69516998 Ki = 0.11 nM T84631 CA49UK 69520512 Ki > 17000 nM T84631 C0KB4O 69641445 Ki > 8000 nM T84631 CO3Z8Y 69654811 Ki > 15000 nM T84631 C6AU1R 70252985 Ki = 840 nM T84631 CTO5I6 70253788 Ki > 3000 nM T84631 C8A7ZJ 70306716 Ki = 45 nM T84631 C0WKD9 70662368 IC50 = 3000 nM T84631 C4IFW3 70683249 Ki = 42 nM T84631 C28CEG 70685001 IC50 = 3 nM T84631 C7U9OA 70687171 IC50 = 80 nM T84631 CN38UY 70687492 Ki = 220 nM T84631 C9EL3C 71260387 Ki = 3660 nM T84631 C28RBT 71449502 IC50 = 3.4 nM T84631 C45SHM 71451304 Ki = 1.5 nM T84631 C15ECT 71451305 IC50 = 2.4 nM T84631 C74KFY 71454853 IC50 = 4 nM T84631 CAM29T 71454854 IC50 = 5.6 nM T84631 C53FKA 71458482 IC50 = 5.4 nM T84631 CX4HG2 71458531 IC50 = 740000 nM T84631 CR1WC4 71461267 IC50 = 6400 nM T84631 C8RPG9 71462026 IC50 = 6.4 nM T84631 CVD3W9 71495381 Ki = 32 nM T84631 CNVH43 71495466 Ki = 170 nM T84631 CA5N2S 71495467 Ki = 260 nM T84631 CQ98NY 71495468 Ki = 1100 nM T84631 CE15GB 71495559 Ki = 3050 nM T84631 CW1Y2L 71495560 Ki = 3200 nM T84631 C5Q9BD 71495561 Ki = 1120 nM T84631 C36MRI 71495659 Ki = 60 nM T84631 C7PDA9 71495660 Ki = 110 nM T84631 CF3C8E 71495661 Ki = 580 nM T84631 CECD13 71495765 Ki = 230 nM T84631 C7LXK1 71495766 Ki = 370 nM T84631 CKQ82B 71495974 Ki = 13900 nM T84631 CSV38K 71495975 Ki = 14100 nM T84631 C7QPA0 71495976 Ki = 16900 nM T84631 CI4P9Z 71495977 Ki = 8890 nM T84631 CE03BA 71496089 Ki = 1200 nM T84631 CLO24G 71496201 Ki = 3410 nM T84631 CIE7A6 71496202 Ki = 2450 nM T84631 CAM0I4 71496204 Ki = 550 nM T84631 CJPF90 71548883 Ki > 9000 nM T84631 C30ZKJ 71561420 Ki = 25000 nM T84631 CH32TL 71561557 Ki = 2510 nM T84631 C83ZNH 71562308 IC50 = 266 ug.mL-1 T84631 C8RW7E 71562631 Ki = 12.3 nM T84631 C4UHB2 71562760 Ki = 415 nM T84631 C0EM6D 71562761 Ki = 237 nM T84631 CNS21T 71562882 Ki = 1260 nM T84631 C3SBE2 71562883 Ki = 8500 nM T84631 C2NY0B 71563006 Ki = 14042 nM T84631 CG46AZ 71563007 Ki = 3700 nM T84631 C2O4SB 71563124 Ki = 9000 nM T84631 C4CT8O 71563125 Ki = 3250 nM T84631 C6I9DJ 71567884 Ki = 650 nM T84631 CC7Z0N 71567885 Ki = 1000 nM T84631 C40CRP 71567886 Ki = 2200 nM T84631 CG8X1C 71567887 Ki > 15000 nM T84631 C5DU6Q 71568014 Ki = 1100 nM T84631 C4ICT8 71568015 Ki = 3700 nM T84631 C9BSO1 71568137 Ki = 290 nM T84631 C9TBN3 71568263 Ki > 15000 nM T84631 CXYQ68 71568403 Ki > 15000 nM T84631 C53BYN 71580813 Ki = 16 nM T84631 C57PCL 71580892 Ki = 1500 nM T84631 CRD4I9 71625797 Ki > 25000 nM T84631 CG1V9P 71627416 Ki > 8000 nM T84631 C9J7NH 71652207 Ki = 5080 nM T84631 CLH52G 71654374 Ki = 2150 nM T84631 C8GDV7 71654376 Ki = 1510 nM T84631 CY29LR 71654530 Ki = 637 nM T84631 C3K6PT 71654532 Ki = 2700 nM T84631 C3X7FP 71654534 Ki = 5190 nM T84631 CCGP56 71654535 Ki = 1960 nM T84631 CZG3Y9 71654536 Ki = 1270 nM T84631 C62ZTJ 71660643 IC50 > 33000 nM T84631 C5D2OL 71698598 Ki = 54400 nM T84631 CGYN76 71698686 Ki = 49300 nM T84631 CD0Z5K 71698687 Ki = 28700 nM T84631 C0DUT2 71698688 Ki = 38200 nM T84631 C60JTA 71698689 Ki = 55600 nM T84631 C35ZJV 71698690 Ki = 111000 nM T84631 C9XSB5 71698770 Ki = 48800 nM T84631 CRN95M 71698771 Ki = 47500 nM T84631 C0LW4G 71698774 Ki = 11200 nM T84631 CH26JR 71698775 Ki = 88200 nM T84631 C0WR9F 71699124 Ki > 100000 nM T84631 CZKL39 71699125 Ki > 100000 nM T84631 C27TZK 71699126 Ki = 34300 nM T84631 CD12FS 71699127 Ki = 25600 nM T84631 CFN7Q4 71699199 Ki = 43000 nM T84631 C7RTF0 71699200 Ki = 62900 nM T84631 C8JE0W 71699201 Ki = 54100 nM T84631 CRAG19 71699203 Ki = 10800 nM T84631 CYAH23 71699286 Ki = 82300 nM T84631 CM8E7F 71699287 Ki = 37000 nM T84631 C9Y3DN 71699288 Ki = 57700 nM T84631 C78DJQ 71711730 IC50 < 10000 nM T84631 CQ3K2V 71719191 Ki = 1803 nM T84631 C4TP1M 71748092 Ki = 1800 nM T84631 CVM7Y6 71748093 Ki = 4400 nM T84631 C8HZ6Q 71748094 Ki = 3700 nM T84631 C6CB0G 71748095 Ki = 3900 nM T84631 C2Z7XJ 71748113 Ki = 3100 nM T84631 CM83VP 72163524 IC50 > 10000 nM T84631 CRBH34 72164200 IC50 > 33000 nM T84631 CWNZ45 72164201 IC50 > 33000 nM T84631 CBVO02 72164443 Ki > 8000 nM T84631 C1W9NH 72164444 Ki > 8000 nM T84631 C6Z3IC 72164445 Ki > 8000 nM T84631 C0CGB5 72164564 Ki > 8000 nM T84631 CN37EY 72164565 Ki = 8200 nM T84631 CIT3O5 72164566 Ki > 8000 nM T84631 C80OFE 72164567 Ki > 8000 nM T84631 CD01PR 72164568 Ki > 8000 nM T84631 C85RCG 72164697 Ki = 7000 nM T84631 CP4M2G 72164698 Ki = 7200 nM T84631 C0EWD8 72164699 Ki = 5600 nM T84631 C9G4PK 72200999 IC50 = 0.5 nM T84631 CG8Z7P 72206621 IC50 = 0.2 nM T84631 CK34ZH 72550138 Ki = 6200 nM T84631 CT45ER 72550807 Ki = 3900 nM T84631 C46TNC 72550811 Ki = 4300 nM T84631 CXM6C2 72550813 Ki = 6650 nM T84631 CLI36U 72551247 Ki = 4000 nM T84631 C7OF4T 72711856 Ki = 57300 nM T84631 C4Z2RL 72711858 Ki > 250000 nM T84631 C14KIG 72711859 Ki = 47100 nM T84631 CN08OJ 72711860 Ki = 91600 nM T84631 C0BCJ7 72711861 Ki = 78000 nM T84631 C4CG6J 72711863 Ki = 63500 nM T84631 C8NCB1 72712043 Ki = 7460 nM T84631 CIO50P 72712044 Ki > 250000 nM T84631 CK4H1G 72712045 Ki = 25100 nM T84631 CDY10L 72712046 Ki = 3830 nM T84631 CH9MT7 72712048 Ki = 23600 nM T84631 CW3QR2 72712049 Ki = 1100 nM T84631 CAL2W7 72712050 Ki = 5640 nM T84631 C2A4TH 72712051 Ki = 6830 nM T84631 CJX7H1 72712052 Ki = 8800 nM T84631 CN73TI 72712053 Ki = 27000 nM T84631 C7W6OH 72712054 Ki = 29600 nM T84631 CT1F6W 72712055 Ki > 250000 nM T84631 CK6BL5 72712056 Ki = 37100 nM T84631 C8L3AV 72712057 Ki = 6310 nM T84631 C6NB1T 72712058 Ki = 6000 nM T84631 C2ZKR0 72712059 Ki = 6730 nM T84631 CZ80WI 72712060 Ki = 7730 nM T84631 C2CBY8 72712061 Ki = 15600 nM T84631 C0U7QR 72712062 Ki = 35100 nM T84631 CB0F1O 72712063 Ki = 48500 nM T84631 CAQ0T5 72712064 Ki = 25000 nM T84631 CS0PO5 72712065 Ki = 36100 nM T84631 CM8QC1 72712066 Ki = 12200 nM T84631 C0YW7A 72712067 Ki = 11100 nM T84631 CHJ25Y 72712068 Ki = 7230 nM T84631 CP4BS0 72712069 Ki = 16400 nM T84631 C3J8RV 72712070 Ki = 606 nM T84631 CQI5T2 72712071 Ki = 37700 nM T84631 COQ58Y 72712072 Ki = 44100 nM T84631 CU4I2F 72712250 Ki = 126000 nM T84631 C64SNL 72712251 Ki = 3720 nM T84631 CI2E4L 72712252 Ki = 133 nM T84631 C9BX1Q 72712253 Ki = 2140 nM T84631 CC73NU 72712254 Ki = 774 nM T84631 CF80WL 72712255 Ki > 250000 nM T84631 CAZ5R4 72725806 Ki = 3000 nM T84631 CPW7T3 72725807 Ki = 57 nM T84631 CM1OK7 72792543 IC50 = 39 nM T84631 CBP05V 72792607 IC50 = 13 nM T84631 CYXT24 72792608 IC50 = 0.6 nM T84631 CO89NF 72792609 IC50 = 0.5 nM T84631 CC50RS 72792610 IC50 = 1 nM T84631 CCEZ71 72792672 IC50 = 3.4 nM T84631 CFRI96 72792673 IC50 = 1.2 nM T84631 C86RTS 72792674 IC50 = 1.4 nM T84631 CI5U3J 72792675 IC50 = 1.4 nM T84631 CQ08NT 72792744 IC50 = 1.9 nM T84631 CWB62R 72792745 IC50 = 2.99 nM T84631 CA8WG3 72792746 IC50 = 1.8 nM T84631 CR17NL 72792747 IC50 = 1.1 nM T84631 CW84BZ 73345684 IC50 = 100 nM T84631 CT21AC 73345685 IC50 = 224 nM T84631 C4FQ0W 73345765 Ki > 6000 nM T84631 CCD54H 73345766 Ki > 6000 nM T84631 CO4A1M 73345767 Ki > 6000 nM T84631 CC2FW1 73345771 Ki > 6000 nM T84631 C3JN8A 73347180 IC50 = 550 nM T84631 CQF46R 73348759 Ki > 6000 nM T84631 CJG30R 73348764 Ki = 4200 nM T84631 CUD26E 73348765 Ki > 6000 nM T84631 CSQ41U 73348767 Ki = 760 nM T84631 C7Y3ZB 73348933 Ki = 88.7 nM T84631 CAJ7O5 73350148 Ki > 1000000 nM T84631 CYL2K9 73350270 IC50 = 167 nM T84631 C1EPR4 73350271 IC50 = 220 nM T84631 CHF47P 73350338 Ki > 6000 nM T84631 C5VP6W 73350339 Ki > 6000 nM T84631 CK45HD 73350340 Ki = 4900 nM T84631 C60BNQ 73350342 Ki > 6000 nM T84631 CL8EG7 73350757 Ki = 2250 nM T84631 C36EPY 73351772 IC50 = 12000 nM T84631 COBX03 73351777 IC50 = 2000 nM T84631 C2NEV3 73351853 Ki > 6000 nM T84631 CX1WJ7 73351856 Ki = 1600 nM T84631 C4CD7U 73351857 Ki > 6000 nM T84631 C69BHN 73353326 Ki > 6000 nM T84631 C26QPS 73353327 Ki > 6000 nM T84631 C7DGZ9 73353328 Ki > 6000 nM T84631 CA2P1B 73353330 Ki > 6000 nM T84631 CPS6J3 73354766 IC50 = 1000 nM T84631 CNRW95 73354848 Ki > 6000 nM T84631 COF2K0 73354849 Ki > 6000 nM T84631 C3VFD6 73354850 Ki = 4300 nM T84631 CL34CV 73354863 Ki > 6000 nM T84631 C5U9CI 73355715 Ki = 0.0042 nM T84631 CXG0B8 73356296 IC50 = 230 nM T84631 C8N4RM 73356390 Ki = 6000 nM T84631 C5MVT3 76310068 Ki = 1200 nM T84631 CH1BJ2 76311085 Ki = 970 nM T84631 C9OKI1 76311087 Ki = 1140 nM T84631 CZU72O 76311088 Ki = 3980 nM T84631 CE3ZI8 76311089 Ki = 6700 nM T84631 C29QNE 76311090 Ki = 4100 nM T84631 C3R8LG 76311091 Ki = 2250 nM T84631 CD4AZ2 76311332 Ki = 769 nM T84631 CSBD17 76314701 Ki = 5810 nM T84631 C6FQ0C 76314925 Ki = 62.2 nM T84631 C9J0BH 76317785 Ki = 9000 nM T84631 C9C4BV 76317871 Ki = 14000 nM T84631 CSY3T8 76318271 Ki = 1940 nM T84631 CI7MO1 76318272 Ki > 15000 nM T84631 C28QGR 76318273 Ki = 6400 nM T84631 C4WUP1 76318274 Ki = 8350 nM T84631 CWZA05 76320988 Ki = 100 nM T84631 C9PJ1H 76321975 Ki = 2060 nM T84631 C7UP8I 76321976 Ki = 641 nM T84631 CP1MR4 76322205 Ki = 21.9 nM T84631 CO28RN 76325189 Ki = 8000 nM T84631 CHNJ05 76325595 Ki = 1100 nM T84631 C6UR1G 76325596 Ki = 24 nM T84631 CDB4R0 76325821 Ki = 62.4 nM T84631 CJ10YI 76328088 IC50 = 3500 nM T84631 C3W5PN 76329159 Ki = 9300 nM T84631 CJ9D8H 76329160 Ki = 880 nM T84631 C6CW8M 76332426 Ki > 43000 nM T84631 CL09IJ 76332819 Ki = 130 nM T84631 CXKG18 76332820 Ki > 15000 nM T84631 CYCA26 76332821 Ki = 1480 nM T84631 CADC95 76336441 Ki = 606 nM T84631 CZ4N5I 76336442 Ki = 1310 nM T84631 C7TNX2 76336443 Ki = 1810 nM T84631 CO54FL 76336676 Ki = 337 nM T84631 C10OJP 76336677 Ki = 1220 nM T84631 CAT95V 76685067 IC50 = 3.41 nM T84631 CMD5V7 86583041 Ki > 9000 nM T84631 CWP85J 87360663 IC50 > 10000 nM T84631 CO6U9I 88582319 Ki = 200 nM T84631 CMC3L7 89399327 Ki = 2610 nM T84631 CKR2A0 90295536 IC50 = 590 nM T84631 C9FDP4 90295556 IC50 = 2510 nM T84631 CM3LT0 90295602 IC50 = 46.64 nM T84631 CSJY38 90295614 IC50 = 57.81 nM T84631 CQ6D0F 90295617 IC50 > 100000 nM T84631 C7OL1W 90295621 IC50 = 130 nM T84631 CD8O6C 90295622 IC50 > 100000 nM T84631 CNOB68 90295624 IC50 = 1220 nM T84631 C9ZC5G 90295630 IC50 = 40.56 nM T84631 C7B6FC 90295663 IC50 = 1860 nM T84631 C8YCR2 90295664 IC50 = 730 nM T84631 CE09FR 90295757 IC50 = 87.17 nM T84631 C97WGT 90295764 IC50 = 190 nM T84631 C6SK4I 90664135 IC50 > 1000 ug.mL-1 T84631 CE60BJ 90664137 IC50 > 1000 ug.mL-1 T84631 CYB39G 90664139 IC50 > 1000 ug.mL-1 T84631 C6KU0A 90664141 IC50 > 1000 ug.mL-1 T84631 C0T4MS 90665251 IC50 > 1000 ug.mL-1 T84631 CD53HR 90665253 IC50 > 1000 ug.mL-1 T84631 C1SAZ8 90666139 Ki = 180 nM T84631 C2ERV8 90666140 Ki = 7070 nM T84631 CSO5R7 90666141 Ki = 4790 nM T84631 C3F0PB 90666142 Ki = 6450 nM T84631 CG1W0R 90666143 Ki = 5520 nM T84631 CI3AX1 90666144 Ki = 51 nM T84631 C43YWM 90666145 Ki = 29 nM T84631 CT45NA 90666146 Ki = 11 nM T84631 C56KQL 90666147 Ki = 20 nM T84631 COH41Y 91666660 Ki = 1400 nM T84631 CUC01L 91799239 Ki = 105 nM T84631 CA90QH 91827690 IC50 = 380 nM T84631 CE28SQ 91972030 IC50 > 100000 nM T84631 CISE50 101353098 IC50 = 7165 nM T84631 C6A3ZK 101886607 Ki = 11600 nM T84631 CTG2Q1 117987029 IC50 = 60.56 nM T84631 C4G7NE 117987044 IC50 = 2210 nM T84631 C3PS6Y 118098650 Ki = 1800 nM T84631 CYH43T 118456915 IC50 > 100000 nM T84631 CM39QL 118456920 IC50 > 100000 nM T84631 C1C3HV 118456930 IC50 > 30000 nM T84631 CKST03 118456931 IC50 = 25000 nM T84631 C4CJM6 118456935 IC50 > 100000 nM T84631 C6EJB5 118456946 IC50 > 100000 nM T84631 C6ZS9A 118456950 IC50 > 100000 nM T84631 CQ43TO 118456975 IC50 = 29000 nM T84631 CL4K5X 118456998 IC50 > 100000 nM T84631 CCR4Y5 118457019 IC50 > 100000 nM T84631 C26CAL 118457021 IC50 > 100000 nM T84631 COY1V8 118457032 IC50 = 22000 nM T84631 CWY2B9 118457044 IC50 = 26000 nM T84631 CS05DP 118457052 IC50 > 100000 nM T84631 CO72PX 118519577 IC50 = 88.53 nM T84631 CFCN48 118519579 IC50 = 20.22 nM T84631 C1FG2P 118519580 IC50 = 1750 nM T84631 C28MKY 118519581 IC50 > 100000 nM T84631 C21COH 118519584 IC50 = 8080 nM T84631 C52CRZ 118519585 IC50 = 74.77 nM T84631 C5X2KG 118519586 IC50 = 25880 nM T84631 CH1ON2 118519588 IC50 > 100000 nM T84631 CVJ3D6 118519593 IC50 = 32.08 nM T84631 CGA28Y 118519594 IC50 = 5530 nM T84631 CH8B3W 118519596 IC50 = 160 nM T84631 CWH39U 118519597 IC50 = 52690 nM T84631 CVEF90 118519598 IC50 = 11360 nM T84631 CZ8N3W 118519604 IC50 > 100000 nM T84631 C3TB4X 118519607 IC50 = 4180 nM T84631 CLE03N 118519608 IC50 = 710 nM T84631 CXK35R 118519612 IC50 > 100000 nM T84631 C46MSP 118542774 Ki = 740 nM T84631 C20WBY 118542785 Ki = 240 nM T84631 CI65YK 118542879 Ki = 200 nM T84631 CEH93P 118542958 Ki = 250 nM T84631 CITU59 118548755 Ki = 750 nM T84631 CMF5R6 118548758 Ki = 850 nM T84631 C1IH2W 118548759 Ki = 1230 nM T84631 C6LZQ3 118548760 Ki = 510 nM T84631 C62ZNW 118548761 Ki = 610 nM T84631 C3WQ9D 118548776 Ki = 1550 nM T84631 CU01RP 118548813 Ki = 660 nM T84631 C2N1YG 118574661 IC50 = 560 nM T84631 CAB58Q 118574662 IC50 = 310 nM T84631 CK75GJ 118574663 IC50 = 37.65 nM T84631 CW82NL 118574664 IC50 = 15770 nM T84631 C3IU6A 118574693 IC50 = 1210 nM T84631 CIU5Z9 118584716 IC50 = 7060 nM T84631 C51RJX 118707613 Ki = 0.32 nM T84631 CM7GL3 118713017 IC50 = 4780 nM T84631 CKS29X 118713018 IC50 = 2.51 nM T84631 CNA91K 118713019 IC50 = 4.89 nM T84631 CV0Y1I 118713020 IC50 = 45.22 nM T84631 C9SK5T 118713021 IC50 = 63.96 nM T84631 CUN3T1 118713022 IC50 = 17.37 nM T84631 C9OU4J 118713023 IC50 = 50.52 nM T84631 C1Z7LV 118713024 IC50 = 20.87 nM T84631 CEJ56B 118713025 IC50 = 1610 nM T84631 CRF62H 118713026 IC50 = 4.71 nM T84631 CY9KW3 118713027 IC50 = 6.59 nM T84631 CRA2J1 118713028 IC50 = 8180 nM T84631 CAS3L5 118713029 IC50 = 5.06 nM T84631 CFHP98 118713030 IC50 = 15.2 nM T84631 CUS29V 118716986 Ki = 18300 nM T84631 C0GRU4 118718129 Ki = 3.1 nM T84631 C3MVG0 118720988 Ki > 8180 nM T84631 C9M2IH 118720990 Ki > 8180 nM T84631 C1E6GW 118720991 Ki > 8180 nM T84631 C9BVI5 118720993 Ki > 8180 nM T84631 C1FQZ6 118720994 Ki > 9000 nM T84631 C0WZA2 118720996 Ki > 8180 nM T84631 CE89KB 118720997 Ki > 8180 nM T84631 CIAL50 118720998 Ki > 8180 nM T84631 C4HLM3 118720999 Ki > 8180 nM T84631 CLD6I3 118721000 Ki > 8180 nM T84631 C0XG7H 118721001 Ki > 8180 nM T84631 CZC53M 118721002 Ki > 8180 nM T84631 C8FZ2L 118721003 Ki > 8180 nM T84631 C0M4IQ 118721004 Ki > 9000 nM T84631 CLRB29 118721005 Ki = 1370 nM T84631 C9B1FX 118721007 Ki > 8180 nM T84631 CRV5Y1 118721008 Ki = 6390 nM T84631 CH6AQ9 118721009 Ki > 8180 nM T84631 CI7YD4 118723652 IC50 = 140 nM T84631 C7ZX1R 118723654 IC50 = 61 nM T84631 CC5L2H 118723655 IC50 = 68 nM T84631 CSE75C 118723704 IC50 = 220 nM T84631 CA41EG 118723706 IC50 = 290 nM T84631 CC52MF 118723708 IC50 = 16 nM T84631 CTF5U9 118723709 IC50 = 3.6 nM T84631 C4U2AW 118723894 IC50 = 352000 nM T84631 CV5JG3 118723904 IC50 = 195000 nM T84631 CP98JL 118723906 IC50 = 229000 nM T84631 C0UO7Q 118723908 IC50 = 344000 nM T84631 C3IA9S 118726913 IC50 = 13 nM T84631 CABH86 118726934 IC50 = 18 nM T84631 COB7H3 118731959 IC50 = 27 nM T84631 CR67JK 118731960 Ki = 90 nM T84631 CMKI65 118731961 IC50 = 298 nM T84631 C4O2IH 118731962 IC50 = 1120 nM T84631 C8OC5Y 118731963 IC50 = 798 nM T84631 C17ARY 118731964 IC50 = 621 nM T84631 CR4O3V 118731965 IC50 = 452 nM T84631 C7Q0EA 118731966 IC50 = 678 nM T84631 CUQ32B 118731967 IC50 = 828 nM T84631 CCV65S 118731968 IC50 = 612 nM T84631 CW5ZV9 118731969 IC50 = 67 nM T84631 CGQW74 118731970 IC50 = 521 nM T84631 CO5X2B 118731971 IC50 = 23 nM T84631 C34UOK 118731972 IC50 = 183 nM T84631 CDX2R9 118731973 IC50 = 286 nM T84631 CYN2A9 118731974 IC50 = 378 nM T84631 C60SWE 118733712 IC50 = 610 nM T84631 C17VDS 118733713 IC50 = 2.01 nM T84631 CWRX39 118733714 IC50 = 1310 nM T84631 C7OU0X 118733715 IC50 = 1420 nM T84631 C1LK8Q 118733716 IC50 = 2620 nM T84631 CN25YW 118733717 IC50 = 2930 nM T84631 CXUG54 118733718 IC50 = 3220 nM T84631 C2YF0P 118733719 IC50 = 3800 nM T84631 COH5X2 118733720 IC50 = 6.58 nM T84631 CO8B5R 118733721 IC50 = 3.25 nM T84631 CV04QG 118733722 IC50 = 2210 nM T84631 C9AVB2 118733723 IC50 = 1830 nM T84631 CU36GW 118733724 IC50 = 1510 nM T84631 C64ALF 118733725 IC50 = 3060 nM T84631 CA8HY2 118733726 IC50 = 5780 nM T84631 CH2EA0 118733727 IC50 = 5320 nM T84631 CKUY41 118733728 IC50 = 10120 nM T84631 CU6F3L 118733729 IC50 = 11020 nM T84631 CY2Z4Q 118733730 IC50 = 10450 nM T84631 CJ5HT0 118733731 IC50 = 11290 nM T84631 C9P2UN 118733732 IC50 = 1870 nM T84631 C0SBJ9 118733733 IC50 = 870 nM T84631 C9YI0Z 118733734 IC50 = 650 nM T84631 CLKN48 118733735 IC50 = 9.46 nM T84631 CQ84KH 118733736 IC50 = 2420 nM T84631 CVYW12 118733737 IC50 = 2720 nM T84631 CW64OQ 118733738 IC50 = 3030 nM T84631 CY0JV9 118733739 IC50 = 3850 nM T84631 CZW8Q0 118733740 IC50 = 3600 nM T84631 CPH87E 118736125 Ki > 62500 nM T84631 C32KLW 118736129 Ki = 12000 nM T84631 CPN2Q3 118736138 Ki = 390 nM T84631 CHQ5P7 118987013 Ki > 9000 nM T84631 CRI9U5 121399126 Ki = 245 nM T84631 CNXI35 121399185 Ki > 28890 nM T84631 CNF2P3 121399230 Ki > 28890 nM T84631 CPHN78 121399237 Ki = 2473 nM T84631 C2TIC0 121399249 Ki > 28890 nM T84631 C3F7RH 121399265 Ki = 340 nM T84631 CV9TX1 121399281 Ki = 2798 nM T84631 C1ZYC9 121399296 Ki = 195 nM T84631 C4Q0HT 121399308 Ki = 544 nM T84631 C2WD1Q 121407246 Ki = 20720 nM T84631 C3WC9Y 121488127 IC50 = 72000 nM T84631 C3YVQ8 122164611 Ki = 850 nM T84631 CY1S5D 122164612 Ki = 900 nM T84631 CKJN32 122164799 IC50 > 30000 nM T84631 CCE7R9 122187957 IC50 = 17.1 nM T84631 CWV2C7 122187958 IC50 = 28.6 nM T84631 CDH51U 122187961 IC50 = 25.9 nM T84631 CT2Q7L 122187963 IC50 = 15.6 nM T84631 CQ2W6H 122187967 IC50 = 6.5 nM T84631 C9KL5N 122192970 Ki = 412 nM T84631 C6SAE8 122192971 Ki = 1010 nM T84631 CZQ6W3 122192972 Ki = 1507 nM T84631 CX7K5B 122192988 Ki = 15160 nM T84631 C1MVP5 122192989 Ki = 1932 nM T84631 CLHV68 122192990 Ki > 28890 nM T84631 CXU4S3 122193791 Ki = 2259 nM T84631 C23NAU 122193792 Ki = 2145 nM T84631 CX79CM 122193793 Ki = 662 nM T84631 C9ASN2 122193794 Ki = 2036 nM T84631 C9Y6SO 122193795 Ki = 28890 nM T84631 CX9T3D 122193796 Ki = 10710 nM T84631 C2FS4M 122193797 Ki = 4227 nM T84631 COMK61 122193798 Ki = 1006 nM T84631 CZL3W8 122193799 Ki = 258 nM T84631 C90QDF 122193800 Ki = 605 nM T84631 CGQA72 122193881 Ki = 378 nM T84631 C9WT4R 122193882 Ki = 246 nM T84631 CSB1Q5 122193883 Ki = 1682 nM T84631 C9BLF1 122193884 Ki = 1553 nM T84631 CM0TS7 122193885 Ki = 1110 nM T84631 CLI82V 122193886 Ki = 1540 nM T84631 CEN5J7 122193887 Ki = 743 nM T84631 CIJ85X 122193888 Ki = 590 nM T84631 C13UCF 122193889 Ki = 518 nM T84631 CJS68F 122193891 Ki = 1748 nM T84631 CTGN19 122193892 Ki = 1416 nM T84631 C62TVJ 122193893 Ki = 3283 nM T84631 CQO8Z9 122193894 Ki = 1082 nM T84631 C9K8SJ 122193895 Ki = 193 nM T84631 C5R8SG 122193896 Ki = 397 nM T84631 C5LR2A 122193897 Ki > 5000 nM T84631 CH2VR6 122193898 Ki = 337 nM T84631 CI6HC5 122193899 Ki = 507 nM T84631 COZP50 122193900 Ki = 257 nM T84631 CH46TB 122194031 Ki = 5315 nM T84631 CGD97N 122194032 Ki = 1035 nM T84631 C6HX9J 122194033 Ki = 234 nM T84631 CN76EH 122194035 Ki = 1053 nM T84631 CU6QD5 122194036 Ki = 409 nM T84631 CR7MG0 122224465 IC50 > 250000 nM T84631 CAI69W 123238067 Ki = 920 nM T84631 C76BAD 123424620 Ki = 180 nM T84631 CK0W2P 127027635 Ki > 9000 nM T84631 CJ6DA9 127028140 IC50 > 10000 nM T84631 CD9KI3 127028141 IC50 > 10000 nM T84631 CPC0M8 127031390 Ki > 9000 nM T84631 CA30BN 127033248 Ki = 25500 nM T84631 CO7PY0 127033521 Ki = 49400 nM T84631 CE0QZ4 127033522 Ki = 22800 nM T84631 C7ZIR9 127034099 Ki = 400 nM T84631 CN4U9B 127037807 IC50 = 51580 nM T84631 C85ROH 127041472 IC50 > 100000 nM T84631 C4T9KU 127045502 Ki = 6800 nM T84631 C4RFP7 127045503 Ki > 13300 nM T84631 C2IOG9 127045504 Ki > 13300 nM T84631 CHK80O 127045505 Ki > 13300 nM T84631 CL6W5N 127045506 Ki > 13300 nM T84631 CE26HW 131955087 IC50 = 71000 nM T84631 CWQ14N 132578544 IC50 = 150 nM T84631 CPSU28 132938122 IC50 = 140 nM T84631 CT2RV6 134130781 IC50 > 1000000 nM T84631 CWV3G6 134131077 IC50 > 200000 nM T84631 CS8FV1 134131084 IC50 > 200000 nM T84631 C92RTL 134131303 IC50 > 200000 nM T84631 CL37SG 134131589 IC50 > 200000 nM T84631 CPQ04R 134132204 Ki > 10000 nM T84631 CC7UO1 134133660 Ki = 1400 nM T84631 C6DPW7 134141496 Ki > 9000 nM T84631 CIRU10 134145163 Ki = 2000 nM T84631 CHA7X9 134146314 Ki = 2500 nM T84631 C9UZI0 134148669 Ki = 3000 nM T84631 CTG65U 134148771 Ki = 1000 nM T84631 CNR48I 134149150 IC50 = 2400 nM T84631 CR6V9U 134150310 Ki = 1050 nM T84631 CNAR93 134150771 IC50 = 1990 nM T84631 C3QEO5 134151811 Ki = 4800 nM T84631 CJZ50O 134153212 IC50 = 2400 nM T84631 CG9UL4 134156593 Ki = 1800 nM T84631 C9JF0Q 134157000 IC50 = 850 nM T84631 CYJ61L 134157128 IC50 = 350 nM T84631 CD06PE 134313025 IC50 = 3800 nM T84631 C6HTD5 135393470 IC50 > 50000 nM T84631 C7NA6E 135393474 IC50 > 50000 nM T84631 CBW03G 135404142 Ki = 810 nM T84631 C8GE5V 135404808 Ki = 8 nM T84631 CD53CZ 135404951 Ki = 0.75 nM T84631 C9YUQ1 135405121 Ki = 0.07 nM T84631 C9SY8U 135406499 Ki = 26 nM T84631 CQEZ96 135406539 Ki = 983 nM T84631 C94GZP 135406646 Ki = 0.31 nM T84631 CP7Z3S 135407592 Ki = 13 nM T84631 C5XA6H 135407717 Ki = 9400 nM T84631 C0OX6T 135407736 Ki = 7800 nM T84631 CA8X0V 135409826 Ki = 3 nM T84631 CD48MU 135415156 Ki = 3.1 nM T84631 CNIE32 135426905 Ki = 0.41 nM T84631 CK1AD7 135426949 Ki = 0.71 nM T84631 C61XOA 135427245 Ki = 16000 nM T84631 CL25SO 135427324 Ki = 8.4 nM T84631 C2I6WX 135430716 Ki = 320 nM T84631 CHMD42 135431470 Ki = 3500 nM T84631 C8WS4O 135443730 Ki = 16000 nM T84631 CTP5V8 135444609 Ki = 2100 nM T84631 C3SMN4 135444666 IC50 = 0.7 nM T84631 C4M5BF 135450980 Ki > 75000 nM T84631 CKA3D2 135451808 Ki = 0.26 nM T84631 C9KLD3 135455964 Ki = 2 nM T84631 CSK06Y 135456121 Ki = 5 nM T84631 CJWC64 135462427 Ki = 3 nM T84631 CXS6B9 135471524 Ki = 5000 nM T84631 C5PO0Q 135471605 Ki = 78 nM T84631 CU8IC7 135474643 Ki = 6 nM T84631 C2PFI8 135475618 Ki = 1300 nM T84631 CI8Z4U 135479981 Ki = 23 nM T84631 C50EKI 135484100 Ki = 0.28 nM T84631 C37PHT 135487779 IC50 = 4.4 nM T84631 CBE9G0 135490854 Ki = 9900 nM T84631 CZGI04 135490911 Ki = 12 nM T84631 C9T1IA 135492878 Ki > 5000 nM T84631 CRNB95 135492887 Ki > 5000 nM T84631 C9TA2B 135501173 Ki = 0.33 nM T84631 CO5UV8 135501194 Ki = 0.43 nM T84631 CMQ6O0 135501618 Ki = 10000 nM T84631 C47UGJ 135503965 Ki = 3 nM T84631 CVA61N 135512760 Ki = 5700 nM T84631 CLO72H 135514651 Ki = 0.42 nM T84631 CP51ZM 135515290 Ki = 0.24 nM T84631 CW7TI2 135515464 Ki = 29 nM T84631 C3MLP1 135517489 Ki = 106 nM T84631 CSW47P 135528873 Ki = 2700 nM T84631 CW9YX8 135530632 Ki = 5.7 nM T84631 CET9Q2 135530746 Ki = 0.5 nM T84631 C4OW8A 135531345 Ki = 0.65 nM T84631 CK97FT 135533257 Ki = 940 nM T84631 CAD75F 135535997 Ki = 30000 nM T84631 C3E4CU 135537603 Ki = 1.2 nM T84631 C67TIA 135544099 IC50 = 2.2 nM T84631 CDT59O 135544137 Ki = 2 nM T84631 CCH49A 135544551 Ki = 890 nM T84631 CKLD47 135544579 Ki = 25000 nM T84631 CSO35D 135546147 Ki = 85 nM T84631 C5RG6Z 135546170 Ki = 2.4 nM T84631 CD9AO5 135548205 Ki = 9 nM T84631 C7Q9YK 135559071 Ki > 150000 nM T84631 CAU8S4 135559072 Ki > 150000 nM T84631 C9D1MQ 135581665 Ki = 44 nM T84631 CB6L5Y 135581668 Ki = 0.1 nM T84631 C5ZFS3 135581673 Ki = 0.34 nM T84631 CYG47F 135581674 Ki = 3 nM T84631 C94JBX 135581677 Ki = 18.5 nM T84631 C05ONT 135581679 Ki = 7.3 nM T84631 CUL71O 135581680 Ki = 0.1 nM T84631 C5YW3X 135581684 Ki = 0.58 nM T84631 CC72AJ 135610111 Ki = 51 nM T84631 C09QFL 135667566 Ki = 10 nM T84631 CR82IN 135677712 Ki = 62 nM T84631 CUX2R7 135677713 Ki = 9.7 nM T84631 C58PSA 135740053 Ki = 1.1 nM T84631 C4VL1K 135740054 Ki = 0.4 nM T84631 CZL58Y 135740055 Ki = 2.2 nM T84631 CR05YT 135740056 Ki = 2 nM T84631 C2O7PT 135740057 Ki = 0.25 nM T84631 C6MZP7 135763271 Ki = 59 nM T84631 C68GTN 135763273 Ki = 61 nM T84631 C91UXW 135802775 Ki = 7 nM T84631 C0AX3J 135802853 Ki = 81 nM T84631 CRB42G 135802854 Ki = 19 nM T84631 CQD2Z1 135855944 Ki = 0.5 nM T84631 C5ZL2K 135857416 IC50 = 1.4 nM T84631 CMJ0B6 135962022 Ki = 58 nM T84631 CUV6M0 135972471 IC50 = 511 nM T84631 CC54EI 135986123 IC50 = 1.5 nM T84631 C9G7TE 135995982 Ki = 10 nM T84631 C78ZVN 136000585 Ki = 1000 nM T84631 CRG5N4 136000680 Ki = 3.162 nM T84631 C1OXJ5 136029174 Ki = 810 nM T84631 C6S5OL 136034781 Ki = 94000 nM T84631 CPSO31 136045813 Ki = 100 nM T84631 CL1K8S 136045814 Ki = 27 nM T84631 C5KO1C 136045815 Ki = 59 nM T84631 C2MDW7 136045816 Ki = 7300 nM T84631 CJIP97 136045817 Ki = 14 nM T84631 C39YHK 136045818 Ki = 7000 nM T84631 CZE5Y4 136045819 Ki = 3700 nM T84631 CT2UQ9 136045820 Ki > 10000 nM T84631 C1S4QD 136045821 Ki = 3500 nM T84631 CYQ70K 136053621 IC50 = 3.5 nM T84631 C46VRO 136058172 Ki = 20 nM T84631 C6Q4FB 136058174 Ki = 37 nM T84631 C34UZI 136058175 Ki = 12 nM T84631 CUX79V 136058176 Ki = 38 nM T84631 CBY56D 136058177 Ki = 254 nM T84631 C4YO6Q 136058178 Ki = 181 nM T84631 CB39EK 136058180 Ki = 51 nM T84631 C8PLB3 136058181 Ki = 88 nM T84631 CSU6X4 136058182 Ki = 184 nM T84631 C0Y3CA 136058183 Ki = 2 nM T84631 C8IH1Z 136058184 Ki = 9 nM T84631 C4LG7S 136058185 Ki = 131 nM T84631 CCX30L 136058186 Ki = 5 nM T84631 C6KG8F 136058187 Ki = 128 nM T84631 CHS25L 136058188 Ki = 19 nM T84631 C8G4TI 136066129 Ki = 0.84 nM T84631 CY6XD7 136066130 Ki = 8.1 nM T84631 CN70IU 136092208 Ki > 75000 nM T84631 C5N3KP 136092209 Ki = 38000 nM T84631 C1BUH6 136092210 Ki = 125000 nM T84631 CFQ2C8 136092211 Ki = 38000 nM T84631 CX5R9J 136092212 Ki = 83000 nM T84631 C35PXN 136092213 Ki = 32000 nM T84631 CEXJ30 136092214 Ki = 41000 nM T84631 CS6QH0 136092215 Ki = 43000 nM T84631 CMR7L4 136092216 Ki = 167000 nM T84631 CN0WR7 136092217 Ki = 13000 nM T84631 COCN35 136092218 Ki = 34000 nM T84631 CA79JC 136092219 Ki = 6800 nM T84631 C5ST7C 136094220 Ki = 20000 nM T84631 CE0JY5 136094222 Ki > 30000 nM T84631 CJ8GD5 136094223 Ki > 30000 nM T84631 CFL8T4 136094224 Ki = 22000 nM T84631 CQW40T 136104458 IC50 > 100000 nM T84631 CI7XJ3 136104459 IC50 > 100000 nM T84631 C5FHI3 136180800 IC50 = 25 nM T84631 CPK6X2 136198635 Ki = 1.5 nM T84631 CRJ5S4 136198636 Ki = 5 nM T84631 C7WE2G 136198637 Ki = 2 nM T84631 C12UWY 136198638 Ki = 3 nM T84631 CT1QN2 136224837 Ki = 89700 nM T84631 CN8BW0 136224847 Ki > 100000 nM T84631 C7KE9J 136224848 Ki > 100000 nM T84631 C7R1TS 136224849 Ki > 100000 nM T84631 CG24CQ 136224854 Ki = 94800 nM T84631 CK4CM2 137028369 Ki > 28890 nM T84631 C3FRZ4 137629177 Ki = 0.034 nM T84631 C6OVC4 137631541 IC50 = 532 nM T84631 C2JT1W 137632528 IC50 = 212000 nM T84631 CL9C4Z 137633250 IC50 = 887 nM T84631 C64QCY 137633331 IC50 = 546000 nM T84631 CTV82J 137635086 IC50 = 127 nM T84631 CZB61A 137635154 IC50 = 165 nM T84631 CSI03M 137635473 IC50 = 243000 nM T84631 C5BOV8 137635960 IC50 = 157 nM T84631 CDQ62V 137637214 Ki > 50000 nM T84631 C9C4IS 137638370 IC50 = 234 nM T84631 C7W4AS 137638513 IC50 > 100000 nM T84631 CI7G6V 137639337 IC50 = 0.00188 ug.mL-1 T84631 C2K8JV 137639385 Ki = 23000 nM T84631 C89DPN 137639579 IC50 = 717 nM T84631 CGT80B 137640248 IC50 > 100000 nM T84631 CZWT21 137640786 IC50 = 360 nM T84631 CKYM10 137641934 IC50 = 354000 nM T84631 CE1XH0 137642026 IC50 = 1.473 ug.mL-1 T84631 C1RG9N 137642543 IC50 = 4065 nM T84631 C7YI0J 137643322 IC50 = 21 nM T84631 CIX05F 137645194 IC50 = 0.00169 ug.mL-1 T84631 CPY2W8 137646429 IC50 = 0.00287 ug.mL-1 T84631 CNO2T8 137647340 IC50 = 505000 nM T84631 C9EO5K 137647755 IC50 = 52000 nM T84631 CA1WS5 137647866 IC50 = 1414 nM T84631 CTJW91 137647903 IC50 = 345 nM T84631 C8RQW5 137647928 IC50 = 78000 nM T84631 CX5PU9 137648045 IC50 = 0.0315 ug.mL-1 T84631 C9F8HU 137648149 IC50 = 0.00527 ug.mL-1 T84631 C37KPL 137648430 IC50 > 100000 nM T84631 CDN2G1 137650387 IC50 = 0.03336 ug.mL-1 T84631 CVC4G9 137652563 IC50 = 42 nM T84631 CTZJ47 137653030 IC50 = 1267 nM T84631 CCH72E 137653236 IC50 = 0.803 ug.mL-1 T84631 CWO52T 137653817 IC50 = 20000 nM T84631 CNX46H 137654508 Ki > 50000 nM T84631 CS0XG8 137654871 IC50 = 113000 nM T84631 C1OXG8 137655944 IC50 = 31000 nM T84631 CG1AP0 137656734 IC50 = 179000 nM T84631 CYEK02 137658233 IC50 > 100000 nM T84631 CL8JG7 137658848 IC50 = 498 nM T84631 CY17AJ 137658996 IC50 = 2212 nM T84631 CYR84Z 137660177 IC50 = 1345 nM T84631 C68LGV 137661693 IC50 = 0.01692 ug.mL-1 T84631 CUZ35A 138115400 IC50 > 100000 nM T84631 CO51HN 139030452 IC50 > 50000 nM T84631 CX07YE 139592452 Ki > 9000 nM T84631 CE6C0A 145970642 Ki = 1940 nM T84631 CVU38Y 145979005 IC50 = 3026 nM T84631 C9QVU2 145981403 IC50 = 81 nM T84631 CZ1R3B 145982984 Ki = 45 nM T84631 CY53BG 145987654 IC50 = 5617 nM T84631 C5ST3M 145987720 IC50 = 1067 nM T84631 C0UIH3 145991316 IC50 = 5735 nM T84631 CM83CB 145993920 IC50 = 8451 nM T84631 C4HLX8 146029523 IC50 > 50000 nM T84631 CSBC71 146680900 IC50 = 31000 nM T84631 CH59QO 155510375 Ki > 100000 nM T84631 CZ28WP 155510611 IC50 = 246 nM T84631 CICU31 155511394 Ki = 28 nM T84631 CZR36C 155511554 IC50 > 100000 nM T84631 C1S8NW 155511576 Ki = 4861 nM T84631 CA81QV 155512709 Ki = 77600 nM T84631 C2VX3G 155512946 Ki > 13300 nM T84631 CTWK05 155513086 Ki = 321 nM T84631 C5K2RF 155513099 IC50 = 272 nM T84631 C52CEV 155513763 IC50 = 981 nM T84631 CZ9S2L 155513899 IC50 = 3189 nM T84631 C2CI8S 155513907 Ki = 15 nM T84631 CYT20V 155514020 Ki > 50000 nM T84631 C4MUP2 155514223 IC50 = 18 nM T84631 CAT98N 155514640 Ki = 460 nM T84631 C37MUL 155515203 IC50 = 3.5 nM T84631 CG9H4N 155515624 Ki = 113900 nM T84631 C7ZM4R 155515728 Ki = 16150 nM T84631 CPUG37 155516479 Ki > 17000 nM T84631 CFRS54 155516565 Ki = 28890 nM T84631 C57VQG 155516820 Ki = 785 nM T84631 CWI23M 155516948 Ki = 9877 nM T84631 CXY80S 155517048 Ki = 4674 nM T84631 C1ZSV0 155517054 Ki = 20480 nM T84631 C7N3OG 155517516 Ki = 20984 nM T84631 CZ7U1E 155517733 IC50 = 315 nM T84631 C5OG8J 155518396 Ki = 211 nM T84631 CF96DM 155518671 Ki = 96000 nM T84631 C4P9BA 155519561 Ki = 20671 nM T84631 C6NX4K 155519661 IC50 = 1584.89 nM T84631 C4MS1B 155519676 IC50 = 63095.73 nM T84631 CEID74 155519809 IC50 = 1079 nM T84631 C7DUX3 155520916 Ki > 100000 nM T84631 CW8JF0 155521080 IC50 = 77 nM T84631 CBA58W 155522743 Ki = 6169 nM T84631 CE01NY 155523107 IC50 > 20000 nM T84631 CSNL72 155523159 IC50 = 6100 nM T84631 CHW08G 155523201 Ki = 2654 nM T84631 CW9K3R 155523263 IC50 > 20000 nM T84631 CGMP07 155523803 IC50 = 260 nM T84631 CH0N9A 155523885 Ki = 7900 nM T84631 C5N4UF 155524709 Ki = 515 nM T84631 C7FXS3 155524763 IC50 = 7900 nM T84631 CYL8M0 155526377 Ki = 104200 nM T84631 CDT90I 155526882 Ki = 4333 nM T84631 C8F0RX 155526963 IC50 = 234 nM T84631 CX7CO2 155527010 Ki = 7400 nM T84631 CES4H0 155527736 Ki = 13342 nM T84631 CN3BH5 155527998 IC50 = 50118.72 nM T84631 CHYW65 155528639 IC50 = 5011.87 nM T84631 CG68UH 155529134 IC50 > 20000 nM T84631 CD7O2G 155530095 IC50 = 63095.73 nM T84631 CA82SM 155530516 Ki = 29 nM T84631 CT0N2L 155530721 IC50 = 18500 nM T84631 C35QWO 155531023 IC50 = 3981.07 nM T84631 CAU5B6 155531331 Ki = 1931 nM T84631 CP8K2J 155531811 Ki = 11530 nM T84631 C0UR8Q 155531991 Ki = 134400 nM T84631 C3AL6D 155533619 IC50 = 10 nM T84631 CY3FE6 155533938 IC50 = 4.8 nM T84631 C6F4JA 155534286 IC50 = 653 nM T84631 C7M2UT 155534310 IC50 = 6500 nM T84631 C2JC8E 155534627 Ki = 360 nM T84631 CN3K2L 155534709 Ki = 10697 nM T84631 CWS27U 155535533 IC50 = 1543 nM T84631 CLZO23 155535564 IC50 = 2087 nM T84631 CIHM01 155535907 Ki > 100000 nM T84631 C12HON 155536142 IC50 = 31622.78 nM T84631 CAK5R1 155536805 Ki = 2636 nM T84631 CGP82O 155536856 IC50 = 1700 nM T84631 C6S1JG 155537077 Ki = 8607 nM T84631 CUD5Y4 155537271 Ki = 2693 nM T84631 C7JMK4 155538439 Ki > 13000 nM T84631 C9QE5N 155538514 Ki > 100000 nM T84631 CD9J2M 155538805 Ki = 1612 nM T84631 CX9Q2L 155539448 IC50 = 45 nM T84631 CRT3D4 155540148 Ki = 50730 nM T84631 CT2VP1 155540521 Ki = 1913 nM T84631 CL90DN 155540666 Ki > 10000 nM T84631 CY6DK3 155540964 IC50 = 1995.26 nM T84631 C4CHR9 155542229 Ki = 188400 nM T84631 CI1G4S 155543248 IC50 = 1387 nM T84631 CY3T7E 155544010 IC50 = 220 nM T84631 C2MDQ4 155544600 Ki = 2875 nM T84631 CT4S3M 155544624 IC50 = 9000 nM T84631 CD9C5J 155545050 Ki = 26433 nM T84631 C4Q8CE 155545465 Ki = 1941 nM T84631 CU52QS 155545897 Ki > 10000 nM T84631 CQ51DI 155546002 IC50 = 2000 nM T84631 CJR8Y9 155546116 IC50 = 20 nM T84631 CLRJ05 155546124 Ki = 10276 nM T84631 CET91Y 155546188 IC50 = 179 nM T84631 CH2S6R 155546346 Ki = 520 nM T84631 CK6IX7 155547422 Ki = 12136 nM T84631 C5MB9R 155547962 IC50 = 10000 nM T84631 C0D5YW 155548172 IC50 > 2000 nM T84631 CLFB25 155548371 IC50 = 31622.78 nM T84631 CSI5J1 155548907 Ki = 201800 nM T84631 C2H3XJ 155549088 Ki = 2492 nM T84631 C8M9HD 155550013 Ki = 4177 nM T84631 CWC8X9 155550748 IC50 > 100000 nM T84631 C5X4OZ 155550860 Ki = 4025 nM T84631 CU9FL4 155551858 Ki > 50000 nM T84631 COM52R 155551892 IC50 = 5011.87 nM T84631 CA5VG2 155552651 Ki = 404500 nM T84631 C5S6HO 155553129 Ki = 47400 nM T84631 CZT5N7 155553153 Ki = 1809 nM T84631 CJ3FI5 155553630 IC50 = 79432.82 nM T84631 CA3W7F 155554002 Ki = 570 nM T84631 C5TV4J 155554082 Ki = 20640 nM T84631 CO60RZ 155555054 Ki = 9253 nM T84631 C82AXQ 155555647 Ki = 1643 nM T84631 CJW0Q5 155555987 Ki = 1974 nM T84631 CV0R8Y 155556453 Ki = 24000 nM T84631 CFU32P 155557286 IC50 = 4700 nM T84631 C3GWK1 155557690 Ki = 1980 nM T84631 CSW48V 155557718 IC50 = 398.11 nM T84631 CXL5D4 155558368 Ki > 100000 nM T84631 C9U2VZ 155558446 IC50 = 17800 nM T84631 CUA52W 155559155 IC50 = 960 nM T84631 CNZ1K5 155559920 Ki = 500 nM T84631 C3R5JK 155561209 IC50 = 7400 nM T84631 C3SXY1 155561904 Ki = 39520 nM T84631 C1EOR9 155561935 Ki = 1023 nM T84631 CX5O7K 155562968 Ki > 15000 nM T84631 C87WSX 155563035 Ki = 5500000 nM T84631 CQ6N8F 155564027 IC50 = 513 nM T84631 CD0OB4 155564213 Ki = 3603 nM T84631 C5I0YM 155564398 IC50 = 24 nM T84631 C2ZSL7 155565147 IC50 = 7200 nM T84631 CV6KA7 155565165 Ki = 9786 nM T84631 CM8XB1 155565537 IC50 = 7943.28 nM T84631 CTF0S7 155566456 Ki = 447 nM T84631 CS6XQ9 155566619 Ki = 18087 nM T84631 CGD4R1 155566743 IC50 = 30 nM T84631 CP4F1U 155567613 Ki > 50000 nM T84631 CEZ8B9 155568406 Ki > 100000 nM T84631 CK0EA2 155568484 Ki = 34400 nM T84631 CVK8X3 44338049 IC50 = 4.6 nM T84631 CY8D1H 54585929 Ki = 1258.93 nM T84631 D00KJP 10322586 Ki = 7 nM T84631 D00QDR 65238 IC50 = 170 nM T84631 D01LCS 447480 Ki = 1500 nM T84631 D01RTU 448763 Ki > 1000000 nM T84631 D02AVL 18376720 Ki = 0.005 nM T84631 D02KKL 1282 Ki = 1 nM T84631 D02PAU 16731825 Ki = 0.21 nM T84631 D02XPB 23646462 Ki = 1200 nM T84631 D02YIW 1794 IC50 > 50000 nM T84631 D03QAQ 9869498 Ki = 0.01 nM T84631 D03ZUM 6917805 IC50 = 1600 nM T84631 D06HOI 44249821 IC50 = 6.5 nM T84631 D06MTX 1506 Ki = 14000 nM T84631 D07HWB 10417809 IC50 = 280 nM T84631 D07IBU 10696098 IC50 > 20000 nM T84631 D07SFI 2332 Ki = 200 nM T84631 D07ZRG 46899577 Ki = 2.4 nM T84631 D0C1TS 44272875 Ki = 674 nM T84631 D0CT8A 23646461 Ki = 39000 nM T84631 D0F6EZ 44436702 Ki > 1000000 nM T84631 D0FV9Y 44453269 IC50 = 6 nM T84631 D0G4LX 46233650 Ki = 583 nM T84631 D0I1UF 14035442 Ki = 450 nM T84631 D0J1CC 11948634 Ki = 11400 nM T84631 D0J1QT 44473100 Ki = 5.2 nM T84631 D0JU9N 6914623 Ki = 0.03 nM T84631 D0K7YL 447476 Ki = 78 nM T84631 D0LX0D 46233193 Ki = 14800 nM T84631 D0M1BF 9803617 Ki = 96 nM T84631 D0M4VZ 10456438 IC50 = 1900 nM T84631 D0MQ6K 10574241 Ki = 80 nM T84631 D0O0GT 44272797 Ki = 192 nM T84631 D0ON2Z 204102 Ki = 0.19 nM T84631 D0P7NY 23661637 IC50 = 100000 nM T84631 D0R5KV 4322 Ki = 0.1 nM T84631 D0R9CH 3400921 Ki = 0.007 nM T84631 D0SP2I 6852210 Ki = 27000 nM T84631 D0V7TH 76328755 Ki > 15000 nM T84631 D0Y4KJ 46233192 Ki = 3700 nM T84631 D0Y5IQ 44255320 IC50 = 10000 nM T84631 D0Y8QU 9869156 IC50 > 2500 nM T84631 D0Y9PH 45486355 Ki = 40000 nM T84631 D0Z2PJ 24859718 Ki = 6000 nM T84631 D0Z2TG 442688 IC50 = 560 nM T90985 D05ICT 132010322 Ki = 1 nM T90985 D0G8BM 16722836 IC50 = 340 nM T90985 D0M2TS 71600087 Ki = 2.2 nM T90985 D0O0LQ 11364421 IC50 = 260 nM T90985 D0PH9I 118693659 Ki = 100 nM T90985 D0ZW4W 46907787 IC50 = 103 nM T90985 D0D3PX 46926350 IC50 = 37000 nM T90985 CNQ59G 719444 IC50 = 68000 nM T90985 CS1EI8 4541508 Ki > 40000 nM T90985 CB45RH 4794457 Ki > 40000 nM T90985 CY71BJ 4800411 Ki = 1400 nM T90985 CHU94T 6484105 IC50 = 140000 nM T90985 C81LRG 9581822 IC50 = 120000 nM T90985 C0BW3Q 11260691 IC50 = 342 nM T90985 CMJ01U 11283298 IC50 = 560 nM T90985 C6ONU5 16251975 Ki > 40000 nM T90985 CP60ON 16258758 Ki = 2400 nM T90985 CE3X0C 16265714 Ki <= 450 nM T90985 C6WU8Z 16414715 IC50 = 130000 nM T90985 CBX53R 16457178 IC50 = 220000 nM T90985 C4TC3X 16722832 IC50 = 230 nM T90985 CGFA68 16822024 Ki = 1100 nM T90985 CVGU58 18536615 IC50 = 13000 nM T90985 C6Y4GF 18536633 IC50 = 18000 nM T90985 CDS15V 18536647 IC50 = 88000 nM T90985 C1C3QM 44269241 IC50 > 250000 nM T90985 C98BLM 49871817 IC50 = 110 nM T90985 CG3PR6 52912222 IC50 = 31622.78 nM T90985 CF8B4E 60498769 IC50 = 100000 nM T90985 CIPN50 71760902 Ki = 110 nM T90985 C5TB9S 77843982 Ki = 140 nM T90985 COZ8S1 78319129 Ki = 490 nM T90985 C4IF8T 78425807 Ki = 0.69 nM T90985 CFE7R3 86270928 Ki = 4.2 nM T90985 CDG13U 86295201 IC50 = 3513 nM T90985 C1W3XP 112499930 IC50 = 2300 nM T90985 C3QJ5L 122181550 IC50 = 31622.78 nM T90985 CD24VL 122187519 IC50 = 25990 nM T90985 CH14FC 127032939 IC50 = 7900 nM T90985 CS4NG8 127033568 IC50 > 100000 nM T90985 CSO7R6 135530212 IC50 = 220000 nM T90985 C5F3LV 135567026 IC50 > 100000 nM T90985 CO71RI 137285009 IC50 = 3082 nM T90985 CS9MR6 137285011 IC50 = 2781 nM T90985 CFXE14 137321203 IC50 = 501.19 nM T90985 CXN4U1 137321204 IC50 = 199.53 nM T90985 CR5FO2 137632087 Ki > 40000 nM T90985 C7F4MJ 137632577 Ki = 230 nM T90985 CA2D8W 137632690 Ki > 40000 nM T90985 C12WYV 137633398 IC50 = 67000 nM T90985 CO08EU 137636712 Ki = 5600 nM T90985 CVK32T 137639306 Ki <= 450 nM T90985 CVQE64 137643147 Ki > 40000 nM T90985 CD8VQ1 137643820 Ki > 40000 nM T90985 CRJ2W3 137644677 IC50 = 2200 nM T90985 C8QO2D 137648257 Ki = 200 nM T90985 CA4WO8 137653484 Ki = 220 nM T90985 CZ1K6N 137654718 Ki = 23000 nM T90985 CVH74T 137655200 Ki = 4700 nM T90985 C1YOL6 137657448 Ki = 200 nM T90985 CPRY31 137661484 IC50 = 87000 nM T90985 CU5N8O 137701509 IC50 = 3500 nM T90985 CYV4O3 138756791 IC50 = 4700 nM T90985 CQ6XB7 139030526 IC50 = 15848.93 nM T90985 CD6U7X 145925666 IC50 = 357.1 nM T90985 CC17DU 145964393 IC50 = 933 nM T90985 CH06LF 145964543 IC50 = 392 nM T90985 CCW5X8 145965219 IC50 = 378 nM T90985 CE4D5F 145966579 IC50 = 1951 nM T90985 CXWZ04 145967512 IC50 = 978 nM T90985 CV83ED 145972103 Ki = 5.9 nM T90985 CN70KV 145972360 IC50 = 289 nM T90985 C2RTO8 145972845 IC50 = 229 nM T90985 C6R2YM 145975649 IC50 = 8468 nM T90985 CTAZ41 145975701 IC50 > 50000 nM T90985 CW56PH 145975703 IC50 = 102 nM T90985 CN4O0K 145976012 IC50 = 750 nM T90985 CR28YS 145976646 IC50 = 245 nM T90985 CVJ61U 145977109 IC50 = 3543 nM T90985 CB9F1X 145977980 IC50 = 369 nM T90985 C0MD9U 145978238 IC50 = 558 nM T90985 C9FIY4 153534005 IC50 > 20000 nM T90985 CFD6H1 155352361 IC50 = 36000 nM T90985 CFK2B1 155352401 IC50 = 110000 nM T90985 C27LFN 155514936 IC50 = 1600 nM T90985 D00XRH 91820725 IC50 = 25118.86 nM T90985 D0F5TZ 91827383 IC50 = 31622.78 nM T90985 D0VC0I 5169 IC50 = 20000 nM T90985 D0Y3OO 11327430 IC50 = 3500 nM T31818 CVPF30 11839482 EC50 = 22000 nM T31818 CM5X2F 59821830 EC50 = 20000 nM T31818 C4RKS8 90665331 EC50 = 17000 nM T31818 CE2SV0 90665332 EC50 = 20000 nM T31818 CU8HX1 90665337 EC50 = 19000 nM T31818 CM87PA 90665339 EC50 = 16000 nM T31818 C9SBM0 90665340 EC50 = 40000 nM T31818 CV03RS 90665341 EC50 = 11000 nM T79747 D05FKU 86280523 IC50 = 2.9 nM T79747 D0J5HR 46926973 IC50 = 0.4 nM T79747 C5R1AG 2155128 IC50 = 157 nM T79747 CO9UQ2 3423911 IC50 = 60 nM T79747 CFL8J3 4786512 IC50 = 15 nM T79747 C7SH6B 4993304 IC50 = 8 nM T79747 CX91ZA 9114840 IC50 = 24 nM T79747 C1Y3XQ 57519544 IC50 = 0.074 nM T79747 CMKO61 86303027 IC50 = 1 nM T79747 C3Y9KN 86303187 IC50 = 2 nM T79747 CS5DT3 86303342 IC50 > 50000 nM T79747 C2EOJ5 86763941 IC50 = 0.5 nM T79747 CNB7A0 86763942 IC50 = 5400 nM T79747 CP9N7S 86764709 IC50 = 0.4 nM T79747 CK6E0W 91810397 IC50 = 12 nM T79747 CWM43E 117668573 IC50 = 33000 nM T79747 CL5OI9 117668598 IC50 = 42 nM T79747 CJ94UW 117668684 IC50 > 50000 nM T79747 C2RS7Z 117668802 IC50 = 40 nM T79747 C5IO0K 117671078 IC50 = 10 nM T79747 CE8SK5 117671214 IC50 = 4 nM T79747 CWL5J8 118174040 IC50 = 12 nM T79747 CS6Y1X 118174075 IC50 = 29 nM T79747 CT24YC 118174086 IC50 = 12 nM T79747 CYAX71 118174089 IC50 = 1 nM T79747 CCK2H9 118174109 IC50 = 67 nM T79747 C12LXT 118174114 IC50 = 8 nM T79747 CF38UC 118174137 IC50 = 29 nM T79747 CKXC27 118174156 IC50 = 15 nM T79747 CZ46TY 118174196 IC50 = 1 nM T79747 CZ3A6L 118174200 IC50 = 72 nM T79747 C7GU0A 118174229 IC50 = 11 nM T79747 CDA16S 118174232 IC50 = 11 nM T79747 CS7ER1 118174312 IC50 = 9 nM T79747 C6E8OG 121237481 IC50 = 0.38 nM T79747 C0FQX3 122192846 IC50 = 5 nM T79747 CF0S3G 122192847 IC50 = 2.2 nM T79747 CMXO16 122192848 IC50 = 0.23 nM T79747 C8V4CD 122192849 IC50 = 188 nM T79747 CE68BP 122192850 IC50 = 164 nM T79747 C8V5YM 122192851 IC50 = 40 nM T79747 C19VFK 122192852 IC50 = 30 nM T79747 C15UAX 122192853 IC50 > 1000 nM T79747 CRBE37 122192854 IC50 > 1000 nM T79747 C36ZXY 122192855 IC50 > 1000 nM T79747 CS34WY 122192856 IC50 > 1000 nM T79747 C1JR4U 122192857 IC50 > 1000 nM T79747 CN4RC0 122192858 IC50 > 1000 nM T79747 CO3KE8 122192859 IC50 > 1000 nM T79747 CCVR74 122192860 IC50 = 2.7 nM T79747 CK4BO2 122192861 IC50 = 485 nM T79747 C5JOZ0 122192862 IC50 = 24 nM T79747 CO2WJ4 122192863 IC50 = 483 nM T79747 CN52YT 122192864 IC50 = 0.96 nM T79747 CI9WG3 122192865 IC50 = 0.67 nM T79747 CV2KN5 122192866 IC50 = 0.53 nM T79747 CV4PZ3 122192867 IC50 = 0.19 nM T79747 C5B2DY 122192868 IC50 = 0.11 nM T79747 CB97PK 122195558 IC50 = 27 nM T79747 CF20MA 122195559 IC50 = 5 nM T79747 C98ECK 122234471 IC50 = 130 nM T79747 CL2MT3 122234472 IC50 = 5 nM T79747 CX6NG2 122234473 IC50 = 689 nM T79747 C2R4UL 122234474 IC50 = 7 nM T79747 C32PNV 122234475 IC50 = 1 nM T79747 C4OW0K 122652940 IC50 = 6 nM T79747 C5I6CL 137635434 IC50 = 15 nM T79747 C0Y9EA 137642070 IC50 = 60 nM T79747 CM43SF 137648320 IC50 = 30 nM T79747 CCEM45 137661947 IC50 = 42 nM T79747 C9T0SR 145976580 IC50 = 710 nM T79591 D0L5WM 2157 IC50 = 650 nM T79591 D0S6JG 5920 Ki = 0.22 nM T79591 D0Z4EI 55245 Ki > 1250 nM T79591 D01QXY 9862248 Ki = 1.09 nM T79591 D03MYO 15981237 EC50 = 3740 nM T79591 D07ZTD 15942005 Ki = 12500 nM T79591 D0J6XC 5803 IC50 = 0.14 nM T79591 D0V5FQ 166559 Ki = 40 nM T79591 D02WGY 10299876 Ki = 9.6 nM T79591 D07EGS 9874938 Ki = 0.51 nM T79591 CLSK17 5804 IC50 = 0.04074 nM T79591 C47GSU 79170 IC50 = 9200 nM T79591 C57HCR 652088 IC50 = 85300 nM T79591 CB6HQ4 656928 IC50 = 15.14 nM T79591 C5T8GU 2249170 IC50 = 18100 nM T79591 CG59SJ 2404806 IC50 = 47700 nM T79591 CJN3P5 4266779 IC50 = 16600 nM T79591 CU1I3O 4652254 IC50 > 100000 nM T79591 CRQ1O4 9819350 Ki = 0.7 nM T79591 C4PCB9 9825337 EC50 = 23 nM T79591 C3MZ1Y 9843007 Ki = 172 nM T79591 CJ6E2M 9847869 Ki = 20 nM T79591 CA27CJ 9862799 IC50 = 128.82 nM T79591 CZ82PF 9863447 EC50 = 4.5 nM T79591 CC64MT 9869395 IC50 = 1600 nM T79591 CZ1U7X 9932398 IC50 = 9.7 nM T79591 CY01RH 9933119 EC50 = 0.38 nM T79591 CHG6L7 9933993 IC50 = 630 nM T79591 C46NXU 9951790 IC50 = 1.4 nM T79591 CX4MZ9 9980722 IC50 = 19 nM T79591 CZ96GN 10030727 IC50 = 88 nM T79591 CJ05DK 10049652 IC50 = 13 nM T79591 CP1R7A 10113366 IC50 = 360 nM T79591 C72HTV 10135986 IC50 = 420 nM T79591 CMY69T 10137392 IC50 = 600 nM T79591 CGE9I7 10151760 Ki = 228 nM T79591 C1Y3FJ 10174187 Ki = 186 nM T79591 CD4SX7 10202877 IC50 = 2600 nM T79591 CNPD04 10216950 Ki = 69.3 nM T79591 CDY6F5 10238439 Ki = 30.5 nM T79591 C1DYU9 10269704 Ki = 147 nM T79591 CJB2E3 10274474 Ki = 3 nM T79591 C7UYX0 10276774 Ki = 2.1 nM T79591 CH5NX1 10279835 Ki = 126 nM T79591 CW26FQ 10287060 Ki = 2.45 nM T79591 CIB52S 10297431 IC50 = 3300 nM T79591 CSC3T4 10299993 IC50 = 616.6 nM T79591 C81BSZ 10309431 Ki = 127 nM T79591 C09IJX 10310671 Ki > 10000 nM T79591 CT13FC 10310672 Ki > 10000 nM T79591 C0VMH3 10321482 IC50 = 5000 nM T79591 C7TGL0 10322653 Ki = 8 nM T79591 CP8O0Q 10455127 IC50 = 101 nM T79591 C3UAD9 10456672 IC50 = 5.4 nM T79591 C5N7BD 10456830 IC50 = 0.1 nM T79591 C34MFS 10457976 IC50 = 62 nM T79591 C4T6ZH 10479778 IC50 = 4.3 nM T79591 CM4ED8 10479779 IC50 = 2.512 nM T79591 CU42IL 10897325 IC50 = 1400 nM T79591 CX2RY1 10904700 EC50 = 0.3 nM T79591 CZ3SX1 10918755 IC50 = 820 nM T79591 CD9G7N 11164881 IC50 = 12882.5 nM T79591 C6OX1A 11209929 IC50 = 160000 nM T79591 CPY31C 11247142 IC50 = 460 nM T79591 CA8Z1T 11281247 IC50 = 1584.89 nM T79591 CY0M1L 11395277 IC50 = 4365.16 nM T79591 C48UZO 11463526 IC50 = 820 nM T79591 C5CZ2Q 11998611 Ki = 12500 nM T79591 CRJ1N9 11999781 Ki = 42.1 nM T79591 C7N4HR 11999783 Ki = 10.3 nM T79591 CW01OG 12001110 EC50 = 330 nM T79591 C1AU0V 13958302 Ki = 8.72 nM T79591 CDB93J 15219550 IC50 = 19200 nM T79591 CDKZ56 15940421 Ki = 143 nM T79591 CM17XO 15941848 Ki = 35.2 nM T79591 C1QZ3U 15941849 Ki = 285 nM T79591 CRK5V2 15941850 Ki = 1416 nM T79591 C7PV1O 15941997 Ki = 18.6 nM T79591 C7BD0S 15941998 Ki = 186 nM T79591 C93MUZ 15942131 Ki = 30.5 nM T79591 CNCW45 15942413 Ki = 28.4 nM T79591 CEQ1J5 15981204 EC50 = 15640 nM T79591 CZEJ29 15981205 EC50 = 12000 nM T79591 C47AYJ 15981206 EC50 = 3280 nM T79591 CRF9T7 15981207 EC50 = 7010 nM T79591 C4XF0E 15981234 EC50 = 390 nM T79591 C7U4OQ 15981235 EC50 = 700 nM T79591 CT9N6B 15981236 EC50 = 210 nM T79591 CTI37Q 15981238 EC50 = 410 nM T79591 CIM62O 15981239 EC50 = 780 nM T79591 CB6UE5 15981240 EC50 = 2750 nM T79591 CL0FG1 15981241 EC50 = 820 nM T79591 C4BU2G 15981272 EC50 = 4290 nM T79591 C5BO7H 15981273 EC50 = 750 nM T79591 CES0V2 15981274 EC50 = 8880 nM T79591 C2SR1B 15981276 EC50 = 14390 nM T79591 CIB52A 15981279 EC50 = 1250 nM T79591 CWK35C 16730429 IC50 = 99 nM T79591 C7G2AM 18415120 Ki = 235 nM T79591 CD0L4R 21110667 Ki = 201 nM T79591 C0AQU8 21110669 Ki = 814 nM T79591 CZI6V2 21110670 Ki = 1366 nM T79591 C47HQO 21110672 Ki = 1645 nM T79591 CV3FE0 21110673 Ki = 429 nM T79591 CCGP69 21110677 Ki = 710 nM T79591 CM0DL5 21110680 Ki > 10000 nM T79591 CHN91T 21110689 Ki = 1431 nM T79591 CHT5Y9 21110691 Ki = 154 nM T79591 C7TN9A 21110692 Ki = 1638 nM T79591 CX5I2A 21636517 IC50 = 71000 nM T79591 CF2X6V 22339458 EC50 = 12 nM T79591 CF2CQ7 22372339 IC50 > 100000 nM T79591 CFV3P7 23635238 IC50 = 3600 nM T79591 CWE74Y 23635239 IC50 = 3000 nM T79591 CM6S4G 23635240 IC50 = 4100 nM T79591 CPR67K 23635363 IC50 = 6300 nM T79591 CI6D4Y 23635365 IC50 = 22600 nM T79591 CAHT12 23635366 IC50 = 16500 nM T79591 C1G2TO 23635477 IC50 = 52900 nM T79591 C17PKJ 23635478 IC50 > 100000 nM T79591 CC3VU5 23635479 IC50 > 100000 nM T79591 CGU3Z0 23635480 IC50 > 100000 nM T79591 C82WJG 23635600 IC50 > 100000 nM T79591 C18SZO 23635729 IC50 = 21600 nM T79591 C7BLC2 23635731 IC50 > 100000 nM T79591 CE6DP7 23635732 IC50 > 100000 nM T79591 CGL6T0 23635852 IC50 > 100000 nM T79591 CK4XI2 23635853 IC50 > 100000 nM T79591 CY80FR 23635854 IC50 > 100000 nM T79591 C7NAV1 23635855 IC50 = 68900 nM T79591 CU81CL 23635857 IC50 > 100000 nM T79591 C31FPX 23635859 IC50 > 100000 nM T79591 CQ2E7G 23642624 IC50 > 100000 nM T79591 CB38IZ 23644731 IC50 = 269.15 nM T79591 CT5QC3 23648079 IC50 = 0.14 nM T79591 CP7SV3 23648080 IC50 = 26 nM T79591 CYU20W 23648081 IC50 = 10 nM T79591 C3V1BH 23648082 IC50 = 83 nM T79591 C1JIZ5 23648083 IC50 = 4.3 nM T79591 C3QR1F 23648084 IC50 = 9.8 nM T79591 C0N2YD 23648085 IC50 = 7.5 nM T79591 C08JWQ 23648086 IC50 = 5.5 nM T79591 C5INJ3 23648087 IC50 = 460 nM T79591 CTJK20 23648089 IC50 = 670 nM T79591 CE4R6V 23648090 IC50 = 1500 nM T79591 C84TAV 23648093 IC50 = 1300 nM T79591 CB7OK8 23648094 IC50 = 370 nM T79591 C45JQX 23648095 IC50 = 500 nM T79591 C80CEB 23648096 IC50 = 480 nM T79591 C1DLP6 23648097 IC50 = 930 nM T79591 C4LY6R 23648098 IC50 = 39000 nM T79591 C4KX5O 23648099 IC50 = 1800 nM T79591 C9N7IR 23648100 IC50 = 69000 nM T79591 CV20UI 23648101 IC50 = 12.88 nM T79591 CIKD57 23648102 IC50 = 240 nM T79591 CV91YT 23648103 IC50 = 1288.25 nM T79591 C5WKV2 23648104 IC50 = 1200 nM T79591 C5V6OQ 23648105 IC50 = 128.82 nM T79591 C91FSP 23648106 IC50 = 18.2 nM T79591 CBD9J5 23648107 IC50 = 39.81 nM T79591 C1SXM0 23648109 IC50 = 123.03 nM T79591 C98FIL 23648110 IC50 = 457.09 nM T79591 C7R2XE 23648111 IC50 = 295.12 nM T79591 CR85SZ 23648112 IC50 = 30.2 nM T79591 CN2YX0 23648113 IC50 = 100 nM T79591 CC69AB 23648114 IC50 = 1047.13 nM T79591 COP12V 23648115 IC50 = 1174.9 nM T79591 CN5T8D 23648116 IC50 = 851.14 nM T79591 C7ON2Q 23648118 IC50 = 812.83 nM T79591 CXTZ50 23648122 IC50 = 123.03 nM T79591 CZ8J0T 23648123 IC50 = 245.47 nM T79591 C12HDM 23648124 IC50 = 50.12 nM T79591 CFA1Y6 23648126 IC50 = 501.19 nM T79591 C35AZQ 23648127 IC50 = 1479.11 nM T79591 CR1S4E 23648128 IC50 = 549.54 nM T79591 C0WY3I 23648129 IC50 = 239.88 nM T79591 CL60SF 23648130 IC50 = 426.58 nM T79591 C72TJZ 23648131 IC50 = 85.11 nM T79591 COL8Q7 23648132 IC50 = 204.17 nM T79591 CNWC43 23648133 IC50 = 281.84 nM T79591 C4SW8I 23648134 IC50 = 229.09 nM T79591 CQ7M3I 23648135 IC50 = 93.33 nM T79591 CQW43F 23648136 IC50 = 95.5 nM T79591 C62YFJ 23648137 IC50 = 18.2 nM T79591 CICP87 23648138 IC50 = 1148.15 nM T79591 CTE1N2 24748569 EC50 > 10000 nM T79591 C5XD8Q 24830528 IC50 = 230 nM T79591 CR2A9H 24830680 IC50 = 5200 nM T79591 CD6EI3 24830686 IC50 = 190 nM T79591 CKDP62 24830833 IC50 = 5200 nM T79591 CO9E2H 24894049 EC50 = 1056 nM T79591 C5BS8M 25149230 Ki = 16 nM T79591 CJ6LC2 25149503 Ki = 61.6 nM T79591 CT0J6H 25149504 Ki = 1165 nM T79591 CFW74J 25149505 Ki = 3296 nM T79591 C5MFE8 25149592 Ki = 303 nM T79591 CLSD47 25149598 Ki = 183 nM T79591 CZP70F 25150124 Ki = 897 nM T79591 C4MT7I 25150127 Ki = 594 nM T79591 C7G5CL 25150225 Ki = 1760 nM T79591 C57AUE 25150325 Ki = 1.84 nM T79591 CLZ86A 25150424 Ki = 3.74 nM T79591 CRW82I 44136896 IC50 = 8200 nM T79591 CQAT73 44186032 IC50 = 5300 nM T79591 CC0YN9 44186033 IC50 > 50000 nM T79591 C7VZI4 44186034 IC50 = 3500 nM T79591 CR1D9P 44186035 IC50 = 4000 nM T79591 CC32IS 44186097 IC50 = 3800 nM T79591 C2MG6T 44186098 IC50 = 22200 nM T79591 C4XV1B 44186099 IC50 = 4300 nM T79591 CFJ0P8 44186100 IC50 > 50000 nM T79591 C31NSX 44186101 IC50 = 3500 nM T79591 CBM5Z6 44186102 IC50 = 3200 nM T79591 CX10SK 44186103 IC50 = 2300 nM T79591 C8TU3K 44186104 IC50 = 1200 nM T79591 CWY0A2 44186168 IC50 = 9300 nM T79591 CO65HR 44186169 IC50 = 3400 nM T79591 C1TU5I 44186170 IC50 = 1400 nM T79591 CC49MP 44186171 IC50 = 7700 nM T79591 C3M4KR 44186172 IC50 = 3000 nM T79591 C4COU6 44186173 IC50 = 600 nM T79591 C40ENX 44186175 IC50 = 14800 nM T79591 CIL71S 44186232 IC50 > 50000 nM T79591 CP1A5G 44186233 IC50 > 50000 nM T79591 C4CMU9 44186234 IC50 > 50000 nM T79591 CM9V8Z 44186235 IC50 = 1900 nM T79591 CDI86U 44186236 IC50 = 1300 nM T79591 C2YL8N 44186237 IC50 = 4800 nM T79591 CYO36K 44186238 IC50 = 19800 nM T79591 CRHL62 44186239 IC50 = 3000 nM T79591 CS2N6F 44186298 IC50 > 50000 nM T79591 CES48R 44186299 IC50 > 50000 nM T79591 C6XEM3 44186300 IC50 > 50000 nM T79591 C35QER 44186301 IC50 = 30900 nM T79591 CREP27 44186302 IC50 > 50000 nM T79591 CPLW35 44186303 IC50 = 6200 nM T79591 C1PFT0 44186305 IC50 = 33300 nM T79591 CA1EV7 44186421 IC50 = 5800 nM T79591 CU64OD 44186422 IC50 = 5400 nM T79591 C9J0YD 44186423 IC50 = 2600 nM T79591 C25UOE 44186424 IC50 = 1100 nM T79591 CX9U3Q 44186425 IC50 = 1900 nM T79591 C0Z9OK 44186469 IC50 = 4700 nM T79591 CTJ1O5 44186470 IC50 = 3700 nM T79591 CN8QS2 44186471 IC50 = 1300 nM T79591 C78TSP 44186472 IC50 = 810 nM T79591 CL17KI 44186473 IC50 = 7100 nM T79591 COL0S6 44186474 IC50 = 4100 nM T79591 C75UOJ 44186475 IC50 = 13400 nM T79591 C1KVH2 44186476 IC50 > 50000 nM T79591 C3SH2I 44186517 IC50 = 1900 nM T79591 C8X1EA 44186518 IC50 = 6300 nM T79591 CS7K3Y 44186519 IC50 = 8400 nM T79591 CHW5K6 44186520 IC50 > 50000 nM T79591 C58YWK 44186521 IC50 > 50000 nM T79591 CJPO14 44186523 IC50 = 6800 nM T79591 C2NPV9 44186562 IC50 = 9800 nM T79591 CYH38F 44186563 IC50 > 50000 nM T79591 CGXM40 44349576 EC50 = 1500 nM T79591 CB1P0S 44396251 Ki > 1250 nM T79591 CHY1C3 44396271 Ki = 1200 nM T79591 C29MBI 44396272 Ki = 1100 nM T79591 C4TQ6N 44396282 Ki = 670 nM T79591 CH2Y3L 44396283 Ki > 1250 nM T79591 CWZB52 44396284 Ki > 1250 nM T79591 CD80LM 44396296 Ki = 790 nM T79591 C6SI5L 44396297 Ki > 1250 nM T79591 CR4H1E 44396316 Ki > 1250 nM T79591 C45LRH 44396317 Ki > 1250 nM T79591 CA8V4G 44396331 Ki > 1250 nM T79591 CA8OB7 44400181 IC50 = 650 nM T79591 C4G9CF 44403605 IC50 = 3605 nM T79591 CW6EH8 44403606 IC50 = 109 nM T79591 C0L3WU 44403607 IC50 = 1538 nM T79591 COU4B6 44403627 IC50 = 48 nM T79591 CVH75N 44403628 IC50 = 125 nM T79591 CTQ48J 44403634 IC50 = 14 nM T79591 C3SZ4I 44408427 EC50 = 83 nM T79591 CDE12F 44408544 EC50 = 4.1 nM T79591 C3TAU6 44408607 IC50 = 251.19 nM T79591 CM27EY 44417461 IC50 = 460 nM T79591 CC9BF0 44433089 IC50 = 168 nM T79591 CP7C9J 44435761 IC50 > 100000 nM T79591 CWG53Q 44435778 IC50 = 60900 nM T79591 CH56GJ 44435779 IC50 = 69600 nM T79591 CB1UR7 44435786 IC50 = 75600 nM T79591 CL3FT4 44445692 IC50 = 125.89 nM T79591 C20LCQ 44445716 IC50 = 2691.53 nM T79591 C1EGS9 44445719 IC50 = 457.09 nM T79591 CHT8I1 44445726 IC50 = 38.02 nM T79591 C9U7HY 44445727 IC50 = 3467.37 nM T79591 C31JKD 44445730 IC50 = 338.84 nM T79591 C0NH4Z 44445731 IC50 = 616.6 nM T79591 CEX30A 44452442 EC50 = 11 nM T79591 CR5SI0 44476535 EC50 > 10000 nM T79591 CD38FN 44567764 EC50 = 222 nM T79591 CV1W9E 44589465 Ki = 378 nM T79591 C9K7HA 45270610 IC50 > 50000 nM T79591 CUD91T 49862248 EC50 > 10000 nM T79591 CM7BY6 53385590 IC50 = 4500 nM T79591 C6Z7WI 60204885 IC50 = 1200 nM T79591 C05ZRG 69428069 Ki = 91.8 nM T79591 CR2M8J 69844039 Ki = 503 nM T79591 C5SRF8 70681735 Ki = 195 nM T79591 C3A0DO 70682526 IC50 = 5600 nM T79591 CLJU20 70682537 IC50 = 430 nM T79591 C2SVR8 70682538 IC50 = 2500 nM T79591 CBVQ29 70683842 Ki = 24.4 nM T79591 CVON79 70683843 Ki = 300 nM T79591 C9R0NB 70683844 Ki = 1246 nM T79591 CG40IU 70684617 IC50 = 1100 nM T79591 CO1MQ8 70684618 IC50 = 1000 nM T79591 CU5VH3 70684619 IC50 = 3200 nM T79591 CARO49 70685018 Ki > 1250 nM T79591 CVK46F 70686763 IC50 = 4700 nM T79591 CWJ6U3 70686764 IC50 = 100 nM T79591 C70SIB 70688836 IC50 = 1100 nM T79591 CLF25D 70690926 IC50 = 1100 nM T79591 CB3ZC2 70690927 IC50 = 300 nM T79591 C6FA0H 70690939 IC50 = 1600 nM T79591 C90XVL 70693065 IC50 = 2400 nM T79591 CC2EK8 70693080 IC50 = 2500 nM T79591 C2WC4V 70695111 IC50 = 3500 nM T79591 C92QMH 70695112 IC50 = 460 nM T79591 CMNE57 70695113 IC50 = 190 nM T79591 CTQ37A 70697163 IC50 = 2600 nM T79591 CLU28H 71461159 EC50 = 18 nM T79591 CL8K9N 71523879 Ki > 10000 nM T79591 CQ0C5S 71523924 Ki > 10000 nM T79591 C8DI5U 71523925 Ki = 6751 nM T79591 CTU1K7 71523963 Ki = 4866 nM T79591 CGHD73 71570928 IC50 = 9600 nM T79591 C49SBQ 71571065 IC50 = 4200 nM T79591 CE06XT 71571066 IC50 = 1900 nM T79591 CR92GT 71571067 IC50 = 1700 nM T79591 CTUC72 71571068 IC50 > 60000 nM T79591 C7UHM3 71571069 IC50 > 60000 nM T79591 C1P5HY 71571070 IC50 > 60000 nM T79591 C4CNP2 71571213 IC50 > 60000 nM T79591 CAV18D 71571215 IC50 > 60000 nM T79591 C97ISQ 71571216 IC50 > 60000 nM T79591 C5ZT9O 71716541 IC50 > 60000 nM T79591 C1TN8C 71716542 IC50 > 60000 nM T79591 CPJ4T2 71716543 IC50 > 60000 nM T79591 CP9B4C 71716544 IC50 > 60000 nM T79591 C4OE3H 71716545 IC50 > 60000 nM T79591 CIJ84X 71716546 IC50 = 29000 nM T79591 C4XL7Z 71716547 IC50 > 60000 nM T79591 C7BMG8 71716548 IC50 > 60000 nM T79591 C8O2NJ 71716549 IC50 > 60000 nM T79591 CA1Q0X 71716550 IC50 > 60000 nM T79591 CM6ZN5 71716551 IC50 > 60000 nM T79591 CX6RH7 71716552 IC50 > 60000 nM T79591 CTI7H2 71716553 IC50 > 60000 nM T79591 C8YEZ6 71716554 IC50 > 60000 nM T79591 CT3D1M 71717145 IC50 > 60000 nM T79591 CSHP85 71717146 IC50 > 60000 nM T79591 C5K3QG 71717147 IC50 > 60000 nM T79591 C6B5DO 71717148 IC50 > 60000 nM T79591 CK0ZQ9 71717149 IC50 > 60000 nM T79591 C96GSC 71717150 IC50 > 60000 nM T79591 C36SFW 71717155 IC50 > 60000 nM T79591 CLR58A 71717156 IC50 > 60000 nM T79591 CN4A9V 71717771 IC50 > 60000 nM T79591 CPLW58 71717772 IC50 > 60000 nM T79591 CIL03B 71717773 IC50 = 44000 nM T79591 C63QLG 71717774 IC50 = 33000 nM T79591 CV0I1H 71717775 IC50 = 33000 nM T79591 CUN4O0 71717776 IC50 > 60000 nM T79591 CSO2X5 71717777 IC50 > 60000 nM T79591 C52BZC 71717778 IC50 > 60000 nM T79591 CIE8V5 71717779 IC50 > 60000 nM T79591 C46ICD 71717780 IC50 > 60000 nM T79591 CPH02C 71718378 IC50 > 60000 nM T79591 COX71E 71718379 IC50 > 60000 nM T79591 CC94QZ 71718380 IC50 = 58000 nM T79591 CG2TH9 71718381 IC50 = 37000 nM T79591 C6G4BT 71718382 IC50 = 32000 nM T79591 CQ8AI1 71718383 IC50 > 60000 nM T79591 C4KOT9 71718386 IC50 > 60000 nM T79591 CH2TV1 71718387 IC50 > 60000 nM T79591 CXO1S7 71718388 IC50 > 60000 nM T79591 CI6AN0 71718985 IC50 > 60000 nM T79591 C5U7IR 71718986 IC50 > 60000 nM T79591 C0CJ8S 71718987 IC50 > 60000 nM T79591 C4KAZ7 71718988 IC50 > 60000 nM T79591 CIN3V1 71718992 IC50 > 60000 nM T79591 CZ3WG5 71718993 IC50 > 60000 nM T79591 CE6X2K 71718994 IC50 > 60000 nM T79591 C1IH2Q 71718995 IC50 > 60000 nM T79591 CN1RW4 71718996 IC50 > 60000 nM T79591 CKA36P 71718997 IC50 > 60000 nM T79591 C8LWP5 71719585 IC50 > 60000 nM T79591 CQ6BL0 71719586 IC50 > 60000 nM T79591 CFO1J2 71719587 IC50 > 60000 nM T79591 CT0DH9 71719588 IC50 > 60000 nM T79591 C3BT7V 71719589 IC50 > 60000 nM T79591 CBY36L 71719590 IC50 > 60000 nM T79591 C5SPB2 71719591 IC50 > 60000 nM T79591 CYNI30 71719592 IC50 > 60000 nM T79591 CJ5O6Q 71719593 IC50 > 60000 nM T79591 C7EKV1 71719594 IC50 > 60000 nM T79591 CB7O4D 71719597 IC50 > 60000 nM T79591 CD98PS 71719598 IC50 > 60000 nM T79591 CQ7U4O 71719599 IC50 > 60000 nM T79591 CXDE81 71719600 IC50 > 60000 nM T79591 CDM58X 71719601 IC50 > 60000 nM T79591 CCV8I1 71719602 IC50 > 60000 nM T79591 CH1EB5 71719603 IC50 > 60000 nM T79591 CX46KH 71719604 IC50 > 60000 nM T79591 C7KER0 71720182 IC50 = 44000 nM T79591 C0DYJ3 71720183 IC50 = 25000 nM T79591 CY4J2C 71720184 IC50 = 29000 nM T79591 C4Z0VS 71720185 IC50 > 60000 nM T79591 C5H0WP 71720186 IC50 > 60000 nM T79591 C9B4SP 71720187 IC50 > 60000 nM T79591 CHFZ51 71720188 IC50 > 60000 nM T79591 C2FM0U 71720189 IC50 > 60000 nM T79591 CUG52N 71720190 IC50 > 60000 nM T79591 CV1US9 71720192 IC50 > 60000 nM T79591 C7X8QB 71720193 IC50 > 60000 nM T79591 CB56IU 71720826 IC50 > 60000 nM T79591 CS5R7G 71720827 IC50 > 60000 nM T79591 CTF8D3 71720828 IC50 > 60000 nM T79591 CZ71PL 71720830 IC50 > 60000 nM T79591 C0Y9CT 71720831 IC50 > 60000 nM T79591 CP0G7O 73054742 EC50 = 450 nM T79591 CBJ8C9 73055020 EC50 = 39 nM T79591 CCO4X8 73055021 EC50 = 180 nM T79591 CZ8RJ5 73055022 EC50 = 100 nM T79591 C36LIJ 73055023 IC50 > 10000 nM T79591 C25DRF 73055024 IC50 = 230 nM T79591 C27TWJ 76313972 IC50 > 30000 nM T79591 CO3KL0 118726602 Ki = 13.45 nM T79591 C45QSH 118726603 Ki = 16.33 nM T79591 CWQE31 118726604 Ki = 7.74 nM T79591 CZOI45 118726605 Ki = 1.09 nM T79591 C1QZ8J 118726606 Ki = 0.35 nM T79591 C0A9JB 118726607 Ki = 2.05 nM T79591 C94RVF 118726608 Ki = 0.38 nM T79591 C8IDF7 118726609 Ki = 2.77 nM T79591 C4KY2I 118726610 Ki = 0.51 nM T79591 CEW5K8 118726611 Ki = 9.98 nM T79591 CM2R8J 118726612 Ki = 36.53 nM T79591 CZM9O6 118726613 Ki = 32.33 nM T79591 CK8RB5 118726614 Ki = 46.55 nM T79591 CJA6K2 118726615 Ki = 89.89 nM T79591 C2J8PF 118726616 Ki = 199.97 nM T79591 CH1FA8 135528521 IC50 = 32 nM T79591 C0FWQ7 135559141 IC50 = 1513.56 nM T79591 CU20KW 135559142 IC50 = 144.54 nM T79591 CW9R4B 135559143 IC50 = 562.34 nM T79591 CCF02H 145964530 IC50 = 8400 nM T79591 C56SHA 145964597 IC50 = 5400 nM T79591 C5H8EZ 145965425 IC50 = 4200 nM T79591 C98CHS 145977976 IC50 = 10100 nM T79591 D01HAZ 23635364 IC50 = 6900 nM T79591 D01NTN 11350323 IC50 = 1096.48 nM T79591 D01WVE 9872203 IC50 = 2200 nM T79591 D02CGG 44435789 IC50 = 39100 nM T79591 D03VOM 3092218 IC50 = 10600 nM T79591 D03XCG 23635367 IC50 = 25800 nM T79591 D05FRX 11153607 IC50 = 700 nM T79591 D05XMM 44186304 IC50 = 16800 nM T79591 D05ZJC 9925361 IC50 = 26000 nM T79591 D06IJW 23635362 IC50 = 4100 nM T79591 D07MAF 21653696 IC50 = 7400 nM T79591 D08BQI 11291923 IC50 = 19952.62 nM T79591 D09XOC 23635858 IC50 = 4200 nM T79591 D0A5XG 10027822 IC50 = 950 nM T79591 D0G7HF 23635860 IC50 = 33200 nM T79591 D0H6BV 24843916 IC50 = 7700 nM T79591 D0I2GK 71212 IC50 = 0.24 nM T79591 D0I7DH 23635476 IC50 = 18900 nM T79591 D0J0MD 23635730 IC50 = 17500 nM T79591 D0Q9ZN 23648092 IC50 = 680 nM T79591 D0U0GY 44435784 IC50 = 23000 nM T79591 D0U9JC 44435785 IC50 = 21400 nM T79591 D0YU9Z 14899645 IC50 = 28100 nM T79591 D0ZX0Y 23635856 IC50 = 16700 nM T25608 D0Q5XX 445580 EC50 = 11700 nM T25608 D0UE9X 5280933 EC50 = 4620 nM T25608 D0EO2C 51049992 Ki = 4.7 nM T25608 D0V1WQ 24857286 EC50 = 1.9 nM T25608 CKRG59 10466 EC50 = 20892.96 nM T25608 CWY93I 37289 EC50 = 18620.87 nM T25608 C80LUR 154005 EC50 = 2190 nM T25608 CXH9K8 169433 EC50 > 100000 nM T25608 CF1W7M 233085 EC50 > 50118.72 nM T25608 CC05OD 561372 EC50 = 457.09 nM T25608 C19ADF 643684 EC50 = 11481.54 nM T25608 CA9GQ6 674995 IC50 = 12882.5 nM T25608 CZN6S9 743974 EC50 > 31622.78 nM T25608 C5IW8B 763016 EC50 = 24600 nM T25608 CK4OG8 797771 EC50 = 16700 nM T25608 C8MF6P 805130 IC50 = 2800 nM T25608 CQE21M 818213 EC50 = 16100 nM T25608 CS4H3F 853224 EC50 = 970 nM T25608 C1M7UY 1201156 EC50 = 16800 nM T25608 C4H7CT 1201222 EC50 = 22600 nM T25608 C1ZC6G 1202260 EC50 = 19000 nM T25608 CAIT59 1622278 EC50 = 3200 nM T25608 CP29AK 1646307 EC50 = 12200 nM T25608 C3HK9O 1855223 EC50 = 15100 nM T25608 C9T2OI 2214962 EC50 = 14500 nM T25608 CDU19P 2233248 IC50 = 5300 nM T25608 CB53NT 2843133 IC50 = 8128.31 nM T25608 CTUP01 3514336 EC50 = 5000 nM T25608 CG62ZB 4671033 IC50 = 10000 nM T25608 CQC0E6 4987566 EC50 = 8200 nM T25608 COT13S 5312743 EC50 > 100000 nM T25608 C7ASQ0 5312744 EC50 > 100000 nM T25608 C5YM6G 5332902 IC50 = 251.19 nM T25608 CMZY13 5353640 EC50 = 240 nM T25608 CED08V 9889284 EC50 > 10000 nM T25608 C13JXE 10131213 EC50 = 1258.93 nM T25608 CNZ5W7 10176767 EC50 > 100000 nM T25608 CZ2TJ7 10266133 EC50 = 8810 nM T25608 C15GQR 10292451 EC50 = 7.2 nM T25608 CN2WQ6 11190525 EC50 = 14 nM T25608 CZ3I5E 11203294 Ki = 16 nM T25608 COJW03 11226058 Ki = 15 nM T25608 CNS3C5 11236925 Ki = 20 nM T25608 CE6P9V 11245322 EC50 = 12.3 nM T25608 CG76JQ 11265145 EC50 = 9332.54 nM T25608 C8FV4O 11271473 Ki = 43 nM T25608 CRB69Z 11316164 EC50 = 288.4 nM T25608 CT68IQ 11327107 EC50 = 49 nM T25608 C3N5JU 11398822 EC50 = 15 nM T25608 CV9HT4 11489259 Ki = 21 nM T25608 CWR98I 11507535 EC50 = 8890 nM T25608 C8D7IB 11674915 EC50 = 6.7 nM T25608 CKV9W3 11739868 EC50 = 562.34 nM T25608 C49KIE 11750823 EC50 = 302 nM T25608 CWC60K 11773976 EC50 = 12.59 nM T25608 CIQ15K 11961321 EC50 = 7.6 nM T25608 CP1Q3H 12002185 Ki = 20 nM T25608 CDG28M 12002201 Ki = 19 nM T25608 C2RG8P 12002202 Ki = 18 nM T25608 CBJ23P 14454530 EC50 > 100000 nM T25608 C8GT5Q 15602772 EC50 = 3.8 nM T25608 CZ2SC0 15603739 EC50 = 61 nM T25608 CIK6A2 15603842 EC50 = 11 nM T25608 CF8Q7T 15603946 EC50 = 16 nM T25608 CHYT81 15603947 EC50 = 65 nM T25608 C9B1IW 15604310 EC50 = 1.3 nM T25608 C4QI2Y 15604434 EC50 = 69 nM T25608 CVT35C 15659412 EC50 = 8000 nM T25608 C59DBZ 15659413 EC50 = 6000 nM T25608 CP0SB8 16110418 EC50 > 10000 nM T25608 C3JYS8 16661950 IC50 = 6300 nM T25608 CECK07 17754443 EC50 = 0.1 nM T25608 CQS7M8 19705952 EC50 = 3500 nM T25608 CX2Z9H 20331242 EC50 = 1000 nM T25608 C5A4VN 20993091 EC50 = 1358 nM T25608 CV2BL0 21322577 EC50 = 2484 nM T25608 C46RPA 22036572 EC50 = 3200 nM T25608 C0M3CA 23082739 EC50 = 35 nM T25608 C1GQ3U 23082789 EC50 = 3500 nM T25608 CQK3G8 23082861 EC50 = 1700 nM T25608 C2DB9E 23082877 EC50 = 20 nM T25608 CPL70G 23083015 Ki = 520 nM T25608 C40SFL 23083189 EC50 = 40 nM T25608 CLPE35 23083190 EC50 = 47 nM T25608 CMYD48 23083193 EC50 = 38 nM T25608 CL26XS 23111666 EC50 = 39 nM T25608 C1HEB2 23111668 EC50 = 28 nM T25608 CPFD82 23111671 EC50 = 180 nM T25608 CTK9V6 23111682 Ki = 18 nM T25608 CC3H7G 23111689 EC50 = 29 nM T25608 C27VQJ 23111693 EC50 = 24 nM T25608 CPOD26 23111694 Ki = 6.9 nM T25608 CHT0Q8 23111704 EC50 = 23 nM T25608 C1JK5B 23111708 EC50 = 1700 nM T25608 CT38PB 23111732 EC50 > 10000 nM T25608 C1L6RM 23111734 EC50 = 28 nM T25608 CT32AF 23111754 EC50 = 540 nM T25608 C29JHR 23111764 Ki > 10000 nM T25608 CPSD80 23111766 EC50 = 33 nM T25608 CRY9S6 23111781 EC50 = 22 nM T25608 CE71HA 23111791 EC50 = 21 nM T25608 CA1OT7 23136315 EC50 = 1100 nM T25608 CE3JI2 23136363 EC50 = 34 nM T25608 CV2HD8 23136401 EC50 = 3837 nM T25608 CD4VG3 23136411 EC50 = 134.9 nM T25608 CW3AM0 23136477 EC50 = 1905.46 nM T25608 CJGL28 23157191 EC50 = 6.3 nM T25608 CS7T9B 23157282 Ki = 18 nM T25608 CXSW42 23157589 EC50 = 520 nM T25608 CTE01K 23159839 EC50 = 2700 nM T25608 CQDI97 23159846 EC50 = 2700 nM T25608 CSO9X7 23159951 EC50 = 530 nM T25608 CTQ53W 23346507 EC50 = 758.58 nM T25608 C54OXK 23642299 EC50 = 16 nM T25608 CIA3X8 23699039 EC50 > 100000 nM T25608 CI2K8W 24825479 EC50 = 50.12 nM T25608 C4UM5N 24825480 EC50 = 398.11 nM T25608 C0JYX7 24825481 EC50 = 1122.02 nM T25608 CATZ28 24825482 EC50 = 16595.87 nM T25608 CI30KR 24825483 EC50 = 3981.07 nM T25608 CY0F4L 24825484 EC50 = 218.78 nM T25608 CCG12J 24825485 EC50 = 39.81 nM T25608 C1IZD5 24825486 EC50 = 501.19 nM T25608 C06XPY 24825487 EC50 = 1584.89 nM T25608 CK91WQ 24825488 EC50 < 31622.78 nM T25608 CI7A0X 24825489 EC50 = 12302.69 nM T25608 CQJV71 24825490 EC50 = 251.19 nM T25608 CF80AP 24825491 EC50 = 794.33 nM T25608 CHX09F 24825492 EC50 = 173.78 nM T25608 C49IJM 24825493 EC50 = 1995.26 nM T25608 CTG8N0 24825494 EC50 = 1995.26 nM T25608 C18UWB 24825495 EC50 = 3981.07 nM T25608 CVT5A0 24825496 EC50 = 3981.07 nM T25608 CJS5P6 24825497 EC50 = 5011.87 nM T25608 CWX6U2 24825498 EC50 = 5011.87 nM T25608 C9YCR5 24825499 EC50 < 31622.78 nM T25608 CBG1E0 24825500 EC50 < 31622.78 nM T25608 C9S8OB 24825501 EC50 < 31622.78 nM T25608 C8WMP2 24825502 EC50 < 31622.78 nM T25608 C2L0ON 24825503 EC50 < 31622.78 nM T25608 C9WHV1 24825504 EC50 < 31622.78 nM T25608 CDZ26M 24825505 EC50 = 1258.93 nM T25608 C37KYZ 24825506 EC50 < 31622.78 nM T25608 CG7E5P 24825507 EC50 < 31622.78 nM T25608 CW0VI4 24825508 EC50 < 31622.78 nM T25608 C56XKE 24825509 EC50 = 97.72 nM T25608 CK12YG 24857285 EC50 = 13 nM T25608 C31OGF 24857375 EC50 = 16 nM T25608 CJ1V3Z 24857376 Ki = 12 nM T25608 CK1E7M 24860552 EC50 = 302 nM T25608 C2L8YX 24897670 EC50 = 3.6 nM T25608 CS8T2B 25109512 EC50 = 21000 nM T25608 C32MTA 25149900 EC50 = 5623.41 nM T25608 CZ39BV 25149901 EC50 = 95.5 nM T25608 CK8IX2 25150011 EC50 = 354.81 nM T25608 C5JO1X 25150012 EC50 = 91.2 nM T25608 CG40IY 25150013 EC50 = 89.13 nM T25608 C3FM2H 25150015 EC50 = 87.1 nM T25608 CE7O1K 25150016 EC50 = 74.13 nM T25608 C61UMS 25150018 EC50 = 3715 nM T25608 CMS8T4 25150113 EC50 = 1096.48 nM T25608 CY51JZ 25150114 EC50 = 512.86 nM T25608 CD25SW 25150117 EC50 = 891.25 nM T25608 C1LDN0 25150118 EC50 = 58.88 nM T25608 CYA5N2 25150119 EC50 = 154.88 nM T25608 CYO95C 25150120 EC50 = 43.65 nM T25608 CQB54I 25150121 EC50 = 107.15 nM T25608 C4B8YC 25261464 EC50 = 1100 nM T25608 C6PAV0 25261467 EC50 = 2100 nM T25608 CJZ51K 25272661 IC50 = 2100 nM T25608 CBXQ30 25766502 EC50 = 18800 nM T25608 C5J3YP 42603138 EC50 = 260 nM T25608 C7SGQ2 44223813 EC50 = 500 nM T25608 CL6SX0 44244518 IC50 = 20 nM T25608 CBKM86 44409608 EC50 < 10000 nM T25608 CYB4F6 44409612 EC50 < 10000 nM T25608 CT5AW0 44409664 EC50 = 48.98 nM T25608 CM5VG7 44409665 EC50 = 39.81 nM T25608 C5YKA3 44409670 EC50 = 100 nM T25608 CDRN85 44409676 EC50 = 14.79 nM T25608 CRJZ90 44409677 EC50 = 6.918 nM T25608 CCY03M 44409690 EC50 = 67.61 nM T25608 CLK8N5 44409695 EC50 < 10000 nM T25608 C9YVL7 44409697 EC50 = 323.59 nM T25608 C3Y8JC 44409698 EC50 = 173.78 nM T25608 CDZ92U 44409699 EC50 = 125.89 nM T25608 C8X0EI 44409702 EC50 = 114.82 nM T25608 C0HB4O 44409703 EC50 = 4.467 nM T25608 CMOF79 44409722 EC50 = 2.455 nM T25608 CO6ZV2 44409728 EC50 = 100 nM T25608 C54KUR 44409729 EC50 = 354.81 nM T25608 CIAY19 44409843 EC50 = 10.96 nM T25608 CU92HA 44409844 EC50 = 66.07 nM T25608 CS6RX1 44409877 EC50 = 51.29 nM T25608 C1IT3N 44409878 EC50 = 12.88 nM T25608 CIKM52 44409883 EC50 = 204.17 nM T25608 CFH0P9 44409906 EC50 = 2041 nM T25608 CR0M8C 44409915 EC50 < 10000 nM T25608 C6NF2X 44409916 EC50 = 58.88 nM T25608 CSO5Z9 44409926 EC50 = 9.12 nM T25608 C5RV8P 44409927 EC50 = 53.7 nM T25608 CP6CR2 44409928 EC50 < 10000 nM T25608 C6EL9I 44409929 EC50 = 144.54 nM T25608 CQ8W9J 44409933 EC50 = 36.31 nM T25608 CK8X5D 44571477 EC50 = 970 nM T25608 CX42DJ 44572033 EC50 = 19 nM T25608 CA3JQ8 44572094 EC50 = 260 nM T25608 CVS9U3 44572096 EC50 < 100 nM T25608 CMO3C5 44572097 EC50 = 10 nM T25608 C5KRH4 44589697 EC50 = 85.11 nM T25608 C0LQS4 44591612 IC50 = 10 nM T25608 C3DOW2 44591613 IC50 = 12 nM T25608 CR35KT 44591627 IC50 = 96 nM T25608 CAK8V6 44591628 IC50 = 2 nM T25608 CCWB82 44591629 IC50 = 3 nM T25608 CWR61H 44591630 IC50 = 29 nM T25608 CP4BC2 44591651 IC50 = 156 nM T25608 CJ03XW 44591652 IC50 = 4 nM T25608 C3ZP1K 44591689 IC50 = 89 nM T25608 CT5X0J 44591690 IC50 = 228 nM T25608 C58MHZ 44591691 IC50 = 119 nM T25608 CKHA83 44591692 IC50 = 13 nM T25608 C8KZF9 44591693 IC50 = 10 nM T25608 C7FR4Z 44591719 IC50 = 10 nM T25608 CJ7L9M 44634022 EC50 = 13182.57 nM T25608 CBZG45 44634023 EC50 = 6025.6 nM T25608 CI4SA8 44634024 EC50 = 295.12 nM T25608 CIA25J 45107281 EC50 = 6.2 nM T25608 CA0B5S 45107282 EC50 = 3.9 nM T25608 C1IYL9 45107307 EC50 = 20 nM T25608 C5IAO0 45107311 EC50 = 5 nM T25608 CJN6F1 45107312 EC50 = 3.7 nM T25608 C16NSP 45107317 EC50 = 12 nM T25608 C4UQ9M 45107318 EC50 = 29 nM T25608 CYQC63 45107320 EC50 = 21 nM T25608 CYL14S 45107323 EC50 = 9.9 nM T25608 CHZ23U 45107324 EC50 = 13 nM T25608 C0AHF2 45107476 EC50 = 5.3 nM T25608 CU35QF 45254027 EC50 = 81 nM T25608 C7PRU9 45377306 EC50 > 30000 nM T25608 C3E9VN 46231386 EC50 = 6451 nM T25608 CP93KX 46232307 EC50 = 10 nM T25608 CZ7U2W 46869922 EC50 = 14 nM T25608 CYTP35 46892131 IC50 > 100000 nM T25608 C8XSB6 51031010 Ki = 39 nM T25608 CC91LO 51349860 EC50 = 300 nM T25608 CP9JN0 51349861 EC50 = 154.88 nM T25608 CW1D0B 51349990 EC50 = 300 nM T25608 CIX80K 51349991 EC50 = 260 nM T25608 CNP73Q 51349992 EC50 = 40 nM T25608 C3UA4P 51349993 EC50 = 45 nM T25608 CXR9O8 51350134 EC50 = 1800 nM T25608 CQHP45 51350135 EC50 = 170 nM T25608 CSU3C9 51350136 EC50 = 170 nM T25608 C7PVZ1 51350137 EC50 = 32 nM T25608 CAS51V 51350138 EC50 = 5.7 nM T25608 C1FC4M 51350139 EC50 = 30 nM T25608 CYUQ87 51350140 EC50 = 30 nM T25608 C5SVW3 51350270 EC50 = 120 nM T25608 CCA03I 51350271 EC50 = 240 nM T25608 C4EGI3 51350272 EC50 = 16.6 nM T25608 CO39YF 51350273 EC50 = 82 nM T25608 CRMT67 51350274 EC50 = 120 nM T25608 CYO4V0 51350404 EC50 = 20 nM T25608 C5IT1B 51350405 EC50 = 30 nM T25608 CIY29U 51350406 EC50 = 19 nM T25608 C7EUM1 51350407 EC50 = 9.9 nM T25608 CFYV70 51351414 EC50 = 320 nM T25608 CQIY23 53248846 IC50 = 12 nM T25608 C9MHR0 53248847 EC50 = 113 nM T25608 C7AI4W 54580132 EC50 = 446.68 nM T25608 C4MOV9 54580624 EC50 = 94 nM T25608 C4U8CJ 54580625 EC50 = 114 nM T25608 C3AYC2 54580626 EC50 = 2820 nM T25608 CB1E0U 54580627 IC50 = 10000 nM T25608 CYT3I8 54581632 EC50 = 970 nM T25608 CBJ8D3 54581633 IC50 = 342 nM T25608 C4YRU1 54582145 EC50 = 69.18 nM T25608 C7W8IE 54582148 EC50 = 6309.57 nM T25608 CS03YA 54582149 EC50 = 524.81 nM T25608 CKV29F 54582150 EC50 = 1071.52 nM T25608 CA3JY5 54582628 IC50 = 36 nM T25608 CXQ1S2 54582629 IC50 = 13 nM T25608 C6XPK4 54582630 EC50 = 108 nM T25608 C9K2AQ 54582631 IC50 = 433 nM T25608 C4HD9E 54583097 EC50 = 3311.31 nM T25608 CU5K1Y 54583098 EC50 = 53.7 nM T25608 CJN07Y 54583099 EC50 = 125.89 nM T25608 CYQK29 54583581 EC50 = 1578 nM T25608 C6K1CE 54583582 EC50 = 51 nM T25608 CS26NZ 54584097 EC50 = 12589.25 nM T25608 C31NYG 54584098 EC50 = 75.86 nM T25608 C2N9LK 54584570 EC50 = 686 nM T25608 CDYZ19 54585039 EC50 = 165.96 nM T25608 CHQ70W 54586010 EC50 = 21379.62 nM T25608 C03CFM 54586011 EC50 = 83.18 nM T25608 C4HWR8 54586484 IC50 = 23 nM T25608 C7A1CM 54586485 IC50 = 211 nM T25608 CKJ67Q 54586486 EC50 = 31 nM T25608 C91ENI 54586982 EC50 = 3630.78 nM T25608 CR4XH7 54586983 EC50 = 2454.71 nM T25608 C2W0GK 54586984 EC50 = 186.21 nM T25608 CXO2A9 54669771 EC50 = 40.74 nM T25608 C7WX2N 54757513 EC50 = 4073.8 nM T25608 CY51XQ 54757514 EC50 = 6165.95 nM T25608 C68IMN 54757515 EC50 = 10964.78 nM T25608 C16BGK 54757516 EC50 = 602.56 nM T25608 C7L8YN 54757517 EC50 = 707.95 nM T25608 C7Y5OB 54757518 EC50 = 660.69 nM T25608 CZ1M3Q 54757519 EC50 > 100000 nM T25608 CGL9J4 54757619 EC50 = 9120.11 nM T25608 CN87XO 54757620 EC50 = 9549.93 nM T25608 CHO24D 54757621 EC50 = 4265.8 nM T25608 CHGX78 54757622 EC50 = 2754.23 nM T25608 CV1L0F 54757623 EC50 = 3890.45 nM T25608 C3TE0M 54757624 EC50 = 251.19 nM T25608 C3BDI6 54757625 EC50 = 75.86 nM T25608 C1IHM9 54757626 EC50 = 1122.02 nM T25608 C4CFX9 54757627 EC50 = 512.86 nM T25608 CT53SC 54757732 EC50 = 524.81 nM T25608 CAN93K 54757733 EC50 = 478.63 nM T25608 C32BGX 54757734 EC50 = 186.21 nM T25608 C83TPD 54757735 EC50 = 1071.52 nM T25608 C2P9QA 54757736 EC50 = 177.83 nM T25608 CJ5UA0 54757737 EC50 = 120.23 nM T25608 CJV75N 54757738 EC50 = 134.9 nM T25608 CME5K8 54757739 EC50 = 316.23 nM T25608 C84XHT 54757829 EC50 = 794.33 nM T25608 CRU9P0 54757830 EC50 = 79.43 nM T25608 CBZ7Q3 54757831 EC50 = 43.65 nM T25608 CD8S9Y 56640072 EC50 < 10 nM T25608 CRN7Q3 56680363 EC50 = 42.66 nM T25608 C04CIX 57325674 EC50 = 69 nM T25608 C0NS2J 57325678 EC50 = 570 nM T25608 CKD80Z 57325840 EC50 = 960 nM T25608 CHW75L 57325841 EC50 = 84 nM T25608 CVKL67 57325842 EC50 = 140 nM T25608 CA7IH2 57325916 EC50 = 510 nM T25608 CU8JI5 57325917 EC50 = 91 nM T25608 C0OS7K 57325919 Ki > 10000 nM T25608 CSQB56 57390187 EC50 = 6200 nM T25608 C36RSI 57390188 EC50 = 240 nM T25608 CE48GA 57391957 EC50 = 900 nM T25608 CLQ37O 57391958 EC50 = 1200 nM T25608 CWE7D8 57391959 EC50 = 27000 nM T25608 CVCZ15 57391960 EC50 = 1200 nM T25608 CG6M0N 57393689 EC50 = 580 nM T25608 C2MPC4 57393690 EC50 = 6700 nM T25608 CH17PJ 57393691 EC50 = 64 nM T25608 C31SBK 57393692 EC50 = 25 nM T25608 C3GD1S 57394144 EC50 = 360 nM T25608 CS5X0U 57395404 EC50 = 1100 nM T25608 C81BDZ 57397248 EC50 = 3200 nM T25608 CDH46R 57398937 EC50 = 120 nM T25608 CKB1R2 57398938 EC50 = 58 nM T25608 C2FH6J 57400636 EC50 = 620 nM T25608 CUGV01 57400637 EC50 = 110 nM T25608 CC5TA0 57402427 EC50 = 180 nM T25608 C9AZJ4 57413287 Ki = 99 nM T25608 CS2CD8 57413288 EC50 = 12 nM T25608 CY7BM5 57413289 EC50 = 15 nM T25608 CQP6Y0 57413290 EC50 = 13 nM T25608 C9R1CF 57413373 EC50 = 4.5 nM T25608 CRP91W 57413375 Ki = 12 nM T25608 CRQ45D 57414267 EC50 = 16 nM T25608 CY6I2L 57414268 Ki = 280 nM T25608 CSOE32 57414401 Ki = 21 nM T25608 CI8O0Z 57414402 EC50 = 18 nM T25608 CFI28H 57414403 Ki = 270 nM T25608 C38LHP 57414404 EC50 = 39 nM T25608 CFT94Q 57414405 EC50 = 22 nM T25608 CYT0J7 57414538 EC50 = 290 nM T25608 C7LIV6 57414539 EC50 = 14 nM T25608 C35ADQ 57414540 EC50 = 17 nM T25608 C21PIC 57414542 Ki = 8.8 nM T25608 CN53WX 57414543 Ki = 12 nM T25608 CCT57F 57414676 Ki = 15 nM T25608 C3FY1L 57414677 Ki = 11 nM T25608 CQ7B5A 57414678 EC50 = 29 nM T25608 C1SAB3 57414679 EC50 = 18 nM T25608 CL0NP8 57414680 EC50 = 19 nM T25608 CY5O1Q 57521702 EC50 = 602.56 nM T25608 CDW9N4 57521808 EC50 = 524.81 nM T25608 CZL1W6 57521809 EC50 = 630.96 nM T25608 CT06GY 57521810 EC50 = 933.25 nM T25608 C9S5CH 57521811 EC50 = 512.86 nM T25608 C2DUX1 57521812 EC50 = 851.14 nM T25608 CD8G6M 57521813 EC50 = 1148.15 nM T25608 CDRW60 57521814 EC50 = 2041.74 nM T25608 C76WSM 57521913 EC50 = 4466.84 nM T25608 C9O0LB 57521914 EC50 = 630.96 nM T25608 CS6B7Q 57521915 EC50 = 3548.13 nM T25608 CV8F2A 57521916 EC50 = 602.56 nM T25608 CBTP21 57521917 EC50 = 109.65 nM T25608 CPZQ75 57521918 EC50 = 407.38 nM T25608 CH9K1N 57521919 EC50 = 954.99 nM T25608 C7PEI1 57705531 EC50 = 680 nM T25608 CEY7A5 57705555 EC50 = 110 nM T25608 C51GWM 57705575 EC50 = 1960 nM T25608 C9KPA0 57705648 EC50 = 790 nM T25608 CT8RL2 57705679 EC50 = 90 nM T25608 CGA5E7 57705719 EC50 = 740 nM T25608 C7K4VJ 57705749 EC50 = 140 nM T25608 CM17AI 57705806 EC50 = 120 nM T25608 CF7V9T 57705838 EC50 = 105 nM T25608 CLY04B 57705851 EC50 = 120 nM T25608 C86ICX 57705863 EC50 = 900 nM T25608 C6D8IA 57705880 EC50 = 76 nM T25608 C9F5IV 57705939 EC50 = 227 nM T25608 C3FY4G 57706009 EC50 = 770 nM T25608 CJ70CQ 57706031 EC50 = 690 nM T25608 CK2O3H 57706032 EC50 = 370 nM T25608 C2SFX9 57706097 EC50 = 1830 nM T25608 C8QR5G 57706220 EC50 = 147 nM T25608 C8OH5L 57706227 EC50 = 68 nM T25608 CBDC31 57706280 EC50 = 90 nM T25608 CF35CK 57706451 EC50 = 1410 nM T25608 CPV92M 57706502 EC50 = 310 nM T25608 CBYZ29 57706588 EC50 = 370 nM T25608 C49KUF 57706620 EC50 = 100 nM T25608 C5PZC7 57706642 EC50 = 420 nM T25608 CM97RW 57706720 EC50 = 2200 nM T25608 C5Z4XH 57706778 EC50 = 13 nM T25608 CTH1L7 57706902 EC50 = 88 nM T25608 CG5EK4 57707025 EC50 = 80 nM T25608 CMNJ56 57707110 EC50 = 93 nM T25608 C6V0SY 57707179 EC50 = 100 nM T25608 CQC7P4 57707214 EC50 = 114 nM T25608 CB9C0R 57787398 EC50 = 380 nM T25608 C68FGV 57839754 EC50 > 30000 nM T25608 C20WOJ 58137077 IC50 = 630.96 nM T25608 CRVQ03 58172957 EC50 = 370 nM T25608 C9T0PH 58172961 EC50 = 23 nM T25608 C01QZR 58172969 EC50 = 63 nM T25608 C70RHJ 58172971 EC50 = 1500 nM T25608 C6UOC4 58172978 EC50 = 98 nM T25608 C3WLT5 58172979 EC50 = 27 nM T25608 CYR85D 58172984 EC50 = 970 nM T25608 CUJ5W2 58172986 EC50 = 31 nM T25608 C57AXW 58172988 EC50 = 3100 nM T25608 CJIL12 58172989 EC50 = 49 nM T25608 C02LMG 58172991 EC50 = 89 nM T25608 CQBS49 58172998 EC50 = 210 nM T25608 CQH03N 58172999 EC50 = 190 nM T25608 CM6J1X 58173000 EC50 = 82 nM T25608 CO6P0D 58173002 EC50 = 12 nM T25608 C3LA7I 58218542 EC50 = 560 nM T25608 C0MKH5 58218551 EC50 = 150 nM T25608 CG8U2O 58218571 EC50 = 190 nM T25608 CM7AS3 58218581 EC50 = 360 nM T25608 C68DGL 58218607 EC50 = 140 nM T25608 CWQU02 58218608 EC50 = 67 nM T25608 CS6W8J 58218630 EC50 = 340 nM T25608 CP60JL 58218638 EC50 = 74 nM T25608 CLEV75 58218640 EC50 = 120 nM T25608 C8U1WQ 58218651 Ki = 35 nM T25608 CR0EU5 58218655 EC50 = 2300 nM T25608 C05QYV 58218671 EC50 = 1700 nM T25608 CC0R5G 58218672 EC50 = 570 nM T25608 C9R0HB 58218673 Ki = 13 nM T25608 C3AH2Y 58218694 EC50 = 74 nM T25608 CU0N5T 58218699 EC50 = 3500 nM T25608 C9SHX4 58218709 Ki = 60 nM T25608 C1YUI5 58218726 EC50 = 82 nM T25608 C19SRZ 58218740 EC50 = 150 nM T25608 CMZL87 58319089 EC50 = 2041.74 nM T25608 CUW17O 58319094 EC50 = 83.18 nM T25608 CAEP71 58319098 EC50 = 123.03 nM T25608 C6BK9A 58319107 EC50 = 1000 nM T25608 C6BEP7 58319118 EC50 = 218.78 nM T25608 CR2V9U 58319121 EC50 = 151.36 nM T25608 C6RF5S 58319126 EC50 = 186.21 nM T25608 CX6YK3 58319127 EC50 = 446.68 nM T25608 CU3T9M 58319134 EC50 = 70.79 nM T25608 CB0FY8 58319135 EC50 = 89.13 nM T25608 CB47WD 58319138 EC50 = 16218.1 nM T25608 CP7CY3 58319139 EC50 = 416.87 nM T25608 CT29VJ 58319142 EC50 = 575.44 nM T25608 CU91ZL 58379717 EC50 = 98 nM T25608 C9O4GC 58379893 EC50 = 212 nM T25608 C7OXV2 58379987 EC50 = 105 nM T25608 C5TH9M 58380220 EC50 = 250 nM T25608 CT09DC 58380255 EC50 = 92 nM T25608 COQ92J 58380284 EC50 = 820 nM T25608 CF4B2G 58380381 EC50 = 150 nM T25608 C6GZ3H 58758896 EC50 = 130 nM T25608 C1B5PX 59132613 EC50 = 120 nM T25608 CVI53W 59132740 EC50 = 400 nM T25608 CACS13 59590781 EC50 = 3.4 nM T25608 CU0K4Q 59590895 EC50 = 6.7 nM T25608 CEOP18 60195036 EC50 = 17.38 nM T25608 CS4X9Y 60195037 EC50 = 14.79 nM T25608 CR9C7I 60195038 EC50 = 9.333 nM T25608 CX30BG 60195039 EC50 = 23.44 nM T25608 C7S3HJ 60195040 EC50 = 17.78 nM T25608 CQLD97 60195125 Ki = 4.365 nM T25608 C9DH3R 66562286 EC50 = 35.48 nM T25608 C16SUO 66562287 EC50 = 81.28 nM T25608 CB75OA 66562288 EC50 = 20 nM T25608 CEK8U4 66562289 EC50 = 37.15 nM T25608 C04XUT 66562385 EC50 = 33.11 nM T25608 CI73FC 66562386 EC50 = 16.98 nM T25608 CH5JZ6 66562387 EC50 = 1445.44 nM T25608 CUI9P3 66562388 EC50 = 1949.84 nM T25608 C7D0FE 66562389 EC50 = 141.25 nM T25608 C1RBT5 66562390 EC50 = 144.54 nM T25608 CD0GO5 66562391 EC50 = 426.58 nM T25608 CI7WO1 66562392 EC50 = 38.02 nM T25608 CAU1G2 66562488 EC50 = 18.2 nM T25608 C9HQ8C 67058186 EC50 = 360 nM T25608 CM5IL7 67058222 EC50 = 13 nM T25608 CF0MW1 67058227 EC50 = 19 nM T25608 CK9N8S 67058273 EC50 = 62 nM T25608 CB8KF5 67058307 EC50 = 13 nM T25608 C6NIF3 67072752 EC50 = 19.95 nM T25608 C1BQH0 67085353 EC50 = 310 nM T25608 C5DMN9 67085761 Ki = 10 nM T25608 C6RZL9 67134965 IC50 = 2454.71 nM T25608 CN28HY 67359903 EC50 = 520 nM T25608 C13YCK 67361692 EC50 = 350 nM T25608 CPM76C 67972848 EC50 = 380 nM T25608 CYE04T 68265494 EC50 = 180 nM T25608 C3TM0C 68674201 EC50 = 330 nM T25608 CV82WY 68676271 EC50 = 190 nM T25608 C9X6PR 70522117 EC50 = 977.24 nM T25608 C61LQJ 70901463 EC50 = 3780 nM T25608 CNI46A 71257551 EC50 = 3 nM T25608 C68XRW 71449361 EC50 = 650 nM T25608 COA43P 71449362 EC50 = 2300 nM T25608 CYTQ78 71449363 EC50 = 2100 nM T25608 CEC1V0 71451164 EC50 = 1900 nM T25608 C0MW1K 71454737 EC50 = 1200 nM T25608 CP2VM5 71456495 EC50 = 2300 nM T25608 C1SNX9 71457285 Ki = 370 nM T25608 CG64XE 71458348 EC50 = 1310 nM T25608 C1AH6B 71460190 EC50 = 1200 nM T25608 CI5W0H 71460255 EC50 = 79 nM T25608 CI3Y2S 71460547 EC50 = 21.88 nM T25608 CF3T9Q 71461901 EC50 = 4000 nM T25608 CMZY24 71562312 EC50 = 1000 nM T25608 CS9BX3 71562313 EC50 = 2290.87 nM T25608 CTM07K 71562314 EC50 = 199.53 nM T25608 CVOS18 71562315 EC50 = 346.74 nM T25608 CY1H3I 71562316 EC50 = 144.54 nM T25608 CF2Y6B 71562317 EC50 = 138.04 nM T25608 C80VUQ 71562421 EC50 = 93.33 nM T25608 C0VXG7 71562422 EC50 = 309.03 nM T25608 CR38OD 71562423 EC50 = 138.04 nM T25608 C47QRK 71562424 EC50 = 524.81 nM T25608 C4OZ6V 71562526 EC50 = 338.84 nM T25608 CRP5U8 71562527 EC50 = 223.87 nM T25608 CJ7UZ1 71562637 EC50 = 95.5 nM T25608 C30LJD 71562638 EC50 = 40.74 nM T25608 CN21ZT 71562639 EC50 = 38.02 nM T25608 C6NV8H 71562640 EC50 = 812.83 nM T25608 C2YW9D 71562641 EC50 = 426.58 nM T25608 C4Y2MH 71562768 EC50 = 467.74 nM T25608 CDG40T 71562769 EC50 = 39.81 nM T25608 CKF3X1 71562770 EC50 = 190.55 nM T25608 C8TFI5 71562771 EC50 = 46.77 nM T25608 CHW16K 71562772 EC50 = 263.03 nM T25608 CY73IA 71562773 EC50 = 35.48 nM T25608 C3R0FO 71575419 EC50 = 13.5 nM T25608 CT1D2M 71612680 EC50 = 74.7 nM T25608 CXO1J4 71612681 EC50 = 73.2 nM T25608 CVN8E3 71612682 EC50 = 74.5 nM T25608 C0JNV8 71612683 EC50 = 54.7 nM T25608 C54LIA 71612684 EC50 > 10000 nM T25608 CE4CA6 71612685 EC50 = 36.4 nM T25608 CSBP81 71612894 EC50 = 105.1 nM T25608 CC41RU 71612895 EC50 = 63.7 nM T25608 CMRT56 71612896 EC50 = 55.9 nM T25608 CR1O3Q 71612897 EC50 = 282 nM T25608 C5S4OZ 71612898 EC50 = 46.5 nM T25608 CGKW10 71613092 EC50 = 67.5 nM T25608 CWM47R 71613093 EC50 = 82.4 nM T25608 CV3DW5 71613094 EC50 = 120.7 nM T25608 C1GF4I 71613095 EC50 = 94.8 nM T25608 CM98GB 71613096 EC50 = 145.2 nM T25608 CG6UJ1 71613311 EC50 = 52.9 nM T25608 C19YZB 71613312 EC50 = 30.1 nM T25608 CJY0H8 71613313 EC50 = 39.3 nM T25608 CYQ0D3 71613314 EC50 = 19.1 nM T25608 C2PX9O 71613315 EC50 = 66.7 nM T25608 CI6FY1 71613316 EC50 = 56.7 nM T25608 C7F9BO 71613515 EC50 = 111.1 nM T25608 CBI53Y 71613516 EC50 = 34.2 nM T25608 C0NPS8 71613517 EC50 = 219.8 nM T25608 CBS8D2 71613518 EC50 = 16 nM T25608 CYD54Q 71613519 EC50 = 190.5 nM T25608 C6O0IM 71613520 EC50 = 11.3 nM T25608 C36PAQ 71613521 EC50 = 30.4 nM T25608 C9L8NQ 71615467 EC50 = 122.6 nM T25608 C85KRA 71615468 EC50 = 56.2 nM T25608 C1F3EO 71615469 EC50 = 205.1 nM T25608 CD2IE1 71615470 EC50 = 125 nM T25608 CID4G7 71615666 EC50 = 65.4 nM T25608 C7G5TN 71615667 EC50 = 35.9 nM T25608 CEI6V4 71615668 EC50 = 38.7 nM T25608 CASF10 71615669 EC50 = 61.6 nM T25608 CXAC53 71615670 EC50 = 88 nM T25608 C8DUF7 71615671 EC50 = 132 nM T25608 C1PR6K 71655225 EC50 = 2137.96 nM T25608 CD6EU4 71655226 EC50 = 2511.89 nM T25608 C3XC7G 71655227 EC50 = 22.39 nM T25608 CJMF15 71655293 EC50 = 74.13 nM T25608 CL7BA0 71715951 EC50 < 100 nM T25608 C8F0DH 71816758 EC50 > 30000 nM T25608 CD15WX 71816759 EC50 > 30000 nM T25608 CN3E6S 71816760 EC50 > 30000 nM T25608 C7KN9H 71816761 EC50 = 1420 nM T25608 CMXI29 71816806 EC50 > 30000 nM T25608 CBLG16 71816808 EC50 = 2130 nM T25608 CD0AY7 73345869 EC50 = 18.2 nM T25608 C75PUZ 73345870 EC50 = 363.08 nM T25608 CQ6N0O 73348895 EC50 = 371.54 nM T25608 CPF43O 73354950 EC50 = 724.44 nM T25608 C68LKC 73356502 EC50 = 1380 nM T25608 CQ7T4B 73356514 EC50 = 616.6 nM T25608 CPMI97 73777069 EC50 > 10000 nM T25608 CC0V2Z 73777085 EC50 > 10000 nM T25608 CIX50H 73777111 EC50 > 10000 nM T25608 C9N7VS 73777135 EC50 > 10000 nM T25608 CH5CY8 73777153 EC50 = 6300 nM T25608 CAW6R9 73777156 EC50 = 2500 nM T25608 C0PV3T 73777174 EC50 > 10000 nM T25608 CEYQ78 73777175 EC50 = 8100 nM T25608 C3Y4IL 73891117 EC50 = 6 nM T25608 CR6D4C 75202601 EC50 = 2830 nM T25608 C0CH3I 75202609 EC50 = 530 nM T25608 CM68XD 75204006 EC50 = 190 nM T25608 C07LQH 75204360 EC50 = 210 nM T25608 CYEG23 75204485 EC50 = 940 nM T25608 C0B2NO 75204487 EC50 = 630 nM T25608 CY20UR 75511297 EC50 = 4000 nM T25608 CG3S0Z 75511298 EC50 = 2390 nM T25608 C2SQU1 75511299 EC50 = 2650 nM T25608 C14SZK 75511301 EC50 = 680 nM T25608 C60CGT 75511302 EC50 = 560 nM T25608 C23EHB 75511303 EC50 = 1070 nM T25608 CN3LD9 75511304 EC50 = 700 nM T25608 CX4OE5 75511305 EC50 > 100000 nM T25608 C14EYX 75511306 EC50 = 2670 nM T25608 CL1AJ5 75511307 EC50 = 1200 nM T25608 C6YA1G 75511308 EC50 = 2570 nM T25608 C6MA0F 75511310 EC50 = 210 nM T25608 CRL8X0 75511312 EC50 = 1260 nM T25608 C1W9FN 75511315 EC50 = 13100 nM T25608 C7WVJ5 75511316 EC50 = 3000 nM T25608 C9AQ8B 75511317 EC50 = 4580 nM T25608 C23YEG 76900387 EC50 = 70 nM T25608 CPT9V0 77845055 EC50 = 110 nM T25608 CI2DU6 82051616 EC50 = 11588 nM T25608 CE36PD 82051652 EC50 > 30000 nM T25608 C54DHY 85470884 EC50 = 3340 nM T25608 C6EZF9 85472225 EC50 = 3000 nM T25608 C4EVX7 85970906 EC50 = 9910 nM T25608 COJ03Z 86280676 IC50 > 100000 nM T25608 CD80NR 86288852 EC50 = 0.6 nM T25608 C86BUC 86803183 EC50 = 47500 nM T25608 CX8JY7 86803185 EC50 = 1110 nM T25608 CNFI50 86803186 EC50 = 610 nM T25608 C1KD7H 86803188 EC50 = 2120 nM T25608 CVYK05 86803191 EC50 = 1600 nM T25608 CA24JF 86803193 EC50 = 300 nM T25608 CWC61R 86803196 EC50 = 1130 nM T25608 CP7N5Z 86803219 EC50 = 30100 nM T25608 CNQ59Y 86803224 EC50 = 58 nM T25608 C0W2IX 86817649 EC50 = 500 nM T25608 CN9LT5 87054900 EC50 > 9950 nM T25608 C3L9RY 87055315 EC50 > 100000 nM T25608 CP17IF 87262743 EC50 = 170 nM T25608 CJC5L7 87265393 EC50 = 310 nM T25608 CB94OM 89671280 EC50 = 4 nM T25608 CT92HE 90150977 EC50 = 600 nM T25608 CA41EH 90151022 EC50 = 5900 nM T25608 CQN0H4 90151023 EC50 = 280 nM T25608 CRMJ40 90151177 EC50 = 620 nM T25608 C8IMX2 90151202 EC50 = 1930 nM T25608 C6P9ZY 90151205 EC50 = 440 nM T25608 CX3UW9 90151222 EC50 = 360 nM T25608 CR7G4A 90151279 EC50 = 6270 nM T25608 CDML50 90151283 EC50 = 370 nM T25608 CJ18OS 90151297 EC50 = 510 nM T25608 CI5MN6 90151309 EC50 = 3620 nM T25608 CH0SL3 90151370 EC50 = 100 nM T25608 CIFE09 90151400 EC50 = 360 nM T25608 C7OB1H 90151428 EC50 = 500 nM T25608 CV2U3J 90151435 EC50 = 190 nM T25608 C6Q9TN 90151464 EC50 = 3060 nM T25608 CEC97K 90151466 EC50 = 250 nM T25608 C2NC7J 90151501 EC50 = 150 nM T25608 CJZ8W9 90151514 EC50 = 450 nM T25608 C1U4ZE 90151518 EC50 = 1340 nM T25608 C76OPC 90151527 EC50 = 800 nM T25608 CQ76FH 90151529 EC50 = 480 nM T25608 C31BQW 90151537 EC50 = 2550 nM T25608 C5U6ES 90151568 EC50 = 1180 nM T25608 CP1N2O 90151624 EC50 = 2610 nM T25608 C3DMG7 90151625 EC50 = 220 nM T25608 CRL0F1 90151652 EC50 = 450 nM T25608 C60MBW 90151763 EC50 = 7680 nM T25608 C0XV1D 90151764 EC50 = 110 nM T25608 CMI35V 90158812 EC50 = 37 nM T25608 C2BMT5 90161101 EC50 = 320 nM T25608 C0YQ8E 90176463 EC50 = 20 nM T25608 C72JKP 90357232 EC50 = 1.1 nM T25608 C6SG0A 90372365 EC50 = 29 nM T25608 C7M3AG 90372458 EC50 = 816 nM T25608 C4J1UE 90372616 EC50 = 5.2 nM T25608 CDJ1R8 90418278 EC50 > 5000 nM T25608 C32NHB 90644286 EC50 = 3.5 nM T25608 C71KBF 90644287 EC50 = 71 nM T25608 CN17FZ 90644288 EC50 = 32 nM T25608 CZ1OL4 90644289 EC50 = 65 nM T25608 CIP4R2 90644290 EC50 = 3.8 nM T25608 CIA9O6 90644291 EC50 = 420 nM T25608 C6LG5C 90644292 EC50 = 130 nM T25608 CSPJ89 90644293 EC50 = 9.3 nM T25608 C0HG4I 90644294 EC50 = 81 nM T25608 C0WX4B 90644295 EC50 = 2500 nM T25608 CKP0Q6 90644296 EC50 = 8.6 nM T25608 CFK6R0 90644297 EC50 = 65 nM T25608 CQG80O 90644298 EC50 = 120 nM T25608 CP06GD 90644299 EC50 = 18 nM T25608 CMUJ41 90644300 EC50 = 10 nM T25608 C0LBC3 90644301 EC50 = 14 nM T25608 C45GPE 90644302 EC50 = 230 nM T25608 CKI2V9 90644303 EC50 = 35 nM T25608 C0T3VY 90644561 EC50 = 36 nM T25608 C8CF7R 90644562 EC50 = 9 nM T25608 CX70OS 90655858 EC50 = 3700 nM T25608 CX9YU2 90655859 EC50 = 30000 nM T25608 C3A6NL 90655860 EC50 = 1.7 nM T25608 C9RXS2 90655861 EC50 = 6 nM T25608 CL0R8E 90655862 EC50 = 19 nM T25608 CYN4H6 90655863 EC50 = 22 nM T25608 C8IDE7 91801188 EC50 = 3 nM T25608 CUX4B6 91809187 EC50 = 11 nM T25608 C5G3BA 91824140 EC50 = 146 nM T25608 CR7B3W 91827421 EC50 = 0.3 nM T25608 CCE0N5 100502467 IC50 = 10715.19 nM T25608 CYH40T 102338889 EC50 > 100000 nM T25608 CR75CZ 117886639 EC50 > 10000 nM T25608 C3ZH8N 118129974 Ki = 63 nM T25608 C09KBW 118129979 EC50 = 9 nM T25608 CBM67L 118129981 Ki = 37 nM T25608 CZ3KB5 118129998 EC50 = 16 nM T25608 C7NV5G 118129999 EC50 = 2 nM T25608 CR54JA 118144953 EC50 = 151 nM T25608 CI9Z2D 118144973 EC50 = 4.5 nM T25608 CQMU81 118144976 EC50 = 64 nM T25608 CYE4A0 118144982 EC50 = 3.9 nM T25608 C8BJP0 118145019 EC50 = 2156 nM T25608 C7DWG9 118145020 EC50 = 90 nM T25608 CM5S0K 118145140 EC50 = 15 nM T25608 CCVR32 118151370 EC50 = 1 nM T25608 CV90BK 118623088 EC50 = 7 nM T25608 C7TG3X 118637972 EC50 = 23 nM T25608 C31JBK 118637973 EC50 = 165 nM T25608 C9SFI2 118637974 EC50 = 133 nM T25608 COM74C 118637996 EC50 = 1.7 nM T25608 CZDG27 118638001 EC50 = 30 nM T25608 CEOL73 118642344 EC50 = 2.6 nM T25608 CTGF27 118642372 EC50 = 19 nM T25608 CV13EP 118642379 EC50 = 56 nM T25608 C5ZQ3O 118642384 EC50 = 16 nM T25608 CJ85CQ 118642390 EC50 = 11 nM T25608 CK83MT 118642391 EC50 = 304 nM T25608 C1X5KI 118719473 EC50 = 121.1 nM T25608 CI0DV6 118719474 EC50 = 389.3 nM T25608 C7IG1W 118719717 EC50 = 153.3 nM T25608 CKJZ70 118719720 EC50 = 92.6 nM T25608 CQWP70 118719721 EC50 = 62.3 nM T25608 CH8TE4 118737971 EC50 = 69 nM T25608 CVB7Z5 118737972 EC50 = 63 nM T25608 C9AJC3 118737973 EC50 = 330 nM T25608 CH9FW6 118737974 EC50 = 2600 nM T25608 CX8ZY4 122184685 EC50 = 160 nM T25608 CXKQ09 122184686 EC50 = 540 nM T25608 CGA1I0 122185431 EC50 = 1700 nM T25608 CVZI02 122185432 EC50 = 3800 nM T25608 CZ01FD 122185433 EC50 = 580 nM T25608 CFC26W 122185434 EC50 = 1600 nM T25608 CTYZ26 122185435 EC50 = 30 nM T25608 CP3Q5Y 122185436 EC50 = 19 nM T25608 C36OFW 122185437 EC50 = 100 nM T25608 C2B7NQ 122185438 EC50 = 53 nM T25608 C1Q4MD 122185439 EC50 = 12 nM T25608 CL96RS 122185440 EC50 = 35 nM T25608 CS14ME 122185441 EC50 = 2100 nM T25608 C7VXS9 122185442 EC50 = 3200 nM T25608 CO6QC0 122185443 EC50 = 65 nM T25608 CBSQ43 122185444 EC50 = 49 nM T25608 CLEG07 122185445 EC50 = 560 nM T25608 C1JIA0 122185446 EC50 = 147 nM T25608 C52AYK 122185447 EC50 = 13 nM T25608 C0O6XU 122185448 EC50 = 7.5 nM T25608 CYP30W 122185449 EC50 = 5600 nM T25608 C7N8QL 122185450 EC50 = 120 nM T25608 C9VCR7 122185451 EC50 = 12 nM T25608 CKDT83 122185452 EC50 = 20 nM T25608 C91JIK 122185453 EC50 = 36 nM T25608 C5JQP9 122189672 EC50 = 135.3 nM T25608 C0ZWI4 122189676 EC50 = 135.9 nM T25608 C4FPH2 122189677 EC50 = 108.2 nM T25608 CXWG24 122189678 EC50 = 148.2 nM T25608 CE5FW3 122189680 EC50 = 115.6 nM T25608 CCI6Q8 122189682 EC50 = 121.7 nM T25608 CE0DI6 122189683 EC50 = 140.3 nM T25608 CQK8F3 122189685 EC50 = 147.6 nM T25608 CHOE31 122189737 EC50 = 132.9 nM T25608 C1WUV9 122193735 EC50 = 49.7 nM T25608 C1ND8B 122193736 EC50 = 65.9 nM T25608 C4IEU5 122193737 EC50 = 105.8 nM T25608 C27TUN 122193742 EC50 = 110.3 nM T25608 CUE3S5 122193743 EC50 = 103.6 nM T25608 CC5P0F 122193972 EC50 = 109.5 nM T25608 C0R5CD 122193975 EC50 = 43.6 nM T25608 C7V5SG 124011385 EC50 = 1100 nM T25608 CT3R2Q 126961699 IC50 = 158.49 nM T25608 C9U2VX 127025284 EC50 = 1150 nM T25608 CNK89Y 127025285 EC50 = 6110 nM T25608 CA5G1S 127025488 EC50 = 7730 nM T25608 C29TMV 127025858 EC50 = 23120 nM T25608 CB1UT6 127025866 EC50 = 21010 nM T25608 CQZB72 127025867 EC50 = 16600 nM T25608 C4-AUG-07 127027011 EC50 = 1890 nM T25608 C1I7VD 127027659 EC50 = 3570 nM T25608 C1EN3G 127027726 EC50 = 19580 nM T25608 C4U3QH 127027727 EC50 = 7420 nM T25608 C7ZM2B 127027728 EC50 = 8510 nM T25608 CYE4J9 127027729 EC50 = 1660 nM T25608 C90UDI 127027730 EC50 = 4110 nM T25608 C9C0LW 127029850 EC50 = 96.7 nM T25608 C06KLU 127029851 EC50 = 123.4 nM T25608 CWDA29 127030344 EC50 = 489.78 nM T25608 CZ6M9F 127030713 EC50 < 100000 nM T25608 CP60IR 127030714 EC50 = 199.53 nM T25608 CQPG95 127030715 EC50 = 416.87 nM T25608 CJLP42 127030730 EC50 = 118.5 nM T25608 C1P2AW 127031001 EC50 = 83.18 nM T25608 CL24TF 127031002 EC50 = 208.93 nM T25608 CMC5G3 127031003 EC50 = 47.86 nM T25608 CN38XB 127031412 EC50 = 34.7 nM T25608 CDC7F8 127031413 EC50 = 61.2 nM T25608 C32GDE 127031569 EC50 = 389.05 nM T25608 C80XOP 127032539 EC50 = 46.9 nM T25608 CS9N8K 127033020 EC50 = 512.86 nM T25608 CM9P3T 127033239 EC50 = 68.5 nM T25608 CFZ6D3 127033352 EC50 = 1445.44 nM T25608 CG8LY9 127033353 EC50 = 1819.7 nM T25608 C2OM9J 127033354 EC50 = 5011.87 nM T25608 C0P8LB 127033514 EC50 = 102 nM T25608 CCI7M6 127033818 EC50 = 73.5 nM T25608 CAEB91 127033820 EC50 = 137.5 nM T25608 CM64PE 127033821 EC50 = 85.6 nM T25608 C45XEQ 127034369 EC50 = 64.8 nM T25608 C0MH3C 127034370 EC50 = 48.7 nM T25608 CIQ4F8 127035471 EC50 = 330 nM T25608 CLF1N9 127035472 EC50 = 190 nM T25608 C8K4EU 127035636 EC50 = 23000 nM T25608 C29TRI 127035637 EC50 = 690 nM T25608 C2IAM9 127035638 EC50 = 410 nM T25608 C8EC9W 127035639 EC50 = 750 nM T25608 C5LUP7 127035667 EC50 = 43 nM T25608 C9RSG1 127035668 EC50 = 48 nM T25608 CE42KC 127035669 EC50 = 58 nM T25608 CQ0PC1 127036747 EC50 = 440 nM T25608 CWX6R0 127036748 EC50 = 112 nM T25608 CX6I0B 127036828 EC50 = 36 nM T25608 CVO35L 127036829 EC50 = 69 nM T25608 CE9U3A 127036959 EC50 = 240 nM T25608 CIA6T8 127036960 EC50 = 97 nM T25608 C3C5IY 127037608 EC50 = 43 nM T25608 CL5D9C 127037633 EC50 = 59 nM T25608 CD51PV 127037664 IC50 > 39810.72 nM T25608 C8WAB2 127038348 IC50 > 39810.72 nM T25608 C8JH5V 127038399 IC50 = 100 nM T25608 C9OGB2 127038400 IC50 = 25.12 nM T25608 C76FOP 127038401 IC50 = 501.19 nM T25608 C9D5FS 127038402 IC50 = 6309.57 nM T25608 CRU1T3 127038403 IC50 = 7.943 nM T25608 C0TQN1 127038708 IC50 = 398.11 nM T25608 CJ1S9P 127039385 IC50 = 501.19 nM T25608 CW5RV4 127039708 IC50 = 398.11 nM T25608 C36LBX 127039747 IC50 > 39810.72 nM T25608 CA7P9J 127039748 IC50 = 794.33 nM T25608 C6U4ZF 127040059 IC50 = 398.11 nM T25608 C9YW8X 127040093 IC50 = 630.96 nM T25608 C84IXF 127040094 IC50 = 398.11 nM T25608 CAC71N 127040095 IC50 = 501.19 nM T25608 CLH0B9 127040096 IC50 = 251.19 nM T25608 C69UFE 127040097 IC50 = 501.19 nM T25608 CM15FR 127040115 IC50 = 12.59 nM T25608 C1XBW9 127040116 IC50 = 316.23 nM T25608 C5PJ0H 127040117 IC50 = 79.43 nM T25608 CVL12W 127040118 IC50 = 398.11 nM T25608 CF17PH 127040388 IC50 = 316.23 nM T25608 C04LHZ 127040432 IC50 = 794.33 nM T25608 C2JGV6 127040433 IC50 = 251.19 nM T25608 CZTY30 127040434 IC50 = 1995.26 nM T25608 C17TPU 127040723 IC50 = 3162.28 nM T25608 C8S1MJ 127040748 IC50 = 1995.26 nM T25608 C17ZDX 127040749 IC50 = 7943.28 nM T25608 CG19JK 127041066 IC50 = 1584.89 nM T25608 C8H1RB 127041988 IC50 = 63.1 nM T25608 CPF9A0 127042378 IC50 = 1584.89 nM T25608 CP46OL 127042379 IC50 = 398.11 nM T25608 CI24WP 127042380 IC50 = 1258.93 nM T25608 CM63NP 127042381 IC50 = 398.11 nM T25608 C8FV9D 127042382 IC50 = 1258.93 nM T25608 C9BI7U 127042383 IC50 = 251.19 nM T25608 CDUJ24 127042700 IC50 = 10000 nM T25608 C4O1HN 127042701 IC50 = 2511.89 nM T25608 CPYF81 127042702 IC50 = 31622.78 nM T25608 C0ZGS6 127042703 IC50 > 39810.72 nM T25608 C9MFE4 127042704 IC50 > 39810.72 nM T25608 C8LYI3 127042705 IC50 > 39810.72 nM T25608 C3PIA4 127042713 IC50 = 630.96 nM T25608 C5O8PQ 127045657 EC50 = 38.9 nM T25608 C7R1DO 127045658 EC50 = 114 nM T25608 CXFL01 127045659 EC50 = 11.1 nM T25608 CU87JB 127045863 EC50 = 9.3 nM T25608 CZ32DO 127045864 EC50 = 24.3 nM T25608 CEF75Q 127045865 EC50 = 25.9 nM T25608 C5LF9Z 127045866 EC50 = 25.2 nM T25608 C0IPA3 127045888 EC50 = 214 nM T25608 CN5A8X 127046662 EC50 = 143 nM T25608 CRD1A3 127046663 EC50 = 90.9 nM T25608 CYQ21F 127046664 EC50 = 102 nM T25608 C4F5VZ 127046665 EC50 = 506 nM T25608 CG62RV 127046666 EC50 = 4980 nM T25608 C9GNL4 127046667 EC50 = 862 nM T25608 CI3YB2 127046834 EC50 = 1930 nM T25608 CH83VC 127046960 EC50 = 24.8 nM T25608 CPH9G8 127046961 EC50 = 12 nM T25608 C6OBJ0 127046962 EC50 = 33.2 nM T25608 CH9GZ7 127047527 EC50 = 15.9 nM T25608 CUL5X1 127047528 EC50 = 22.9 nM T25608 CY0E9S 127047529 EC50 = 53.1 nM T25608 CK2G8P 127047530 EC50 = 69.1 nM T25608 C64BKX 127047531 EC50 = 96.7 nM T25608 CWR93I 127047532 EC50 = 79.2 nM T25608 CM65EC 127047533 EC50 = 89.3 nM T25608 C6OPM1 127048827 EC50 = 1280 nM T25608 CH9S7P 127048842 EC50 = 760 nM T25608 CN28RD 127048843 EC50 = 1690 nM T25608 CBTU60 127048844 EC50 = 17940 nM T25608 CZ95XB 127049161 EC50 = 1770 nM T25608 C34HEA 127049498 EC50 = 10620 nM T25608 C8B4QX 127050768 EC50 = 1190 nM T25608 CC3GP9 127050769 EC50 = 4680 nM T25608 C6V3FP 127050770 EC50 = 580 nM T25608 CY1MN8 127050771 EC50 = 4300 nM T25608 CDJ7N9 127051302 EC50 = 1060 nM T25608 C7URZ3 127051657 EC50 > 10000 nM T25608 CE94RI 127051658 EC50 = 580 nM T25608 C9VUY6 127051659 EC50 = 6640 nM T25608 CE6J4T 127051660 EC50 = 1520 nM T25608 C5AJR9 127051855 EC50 > 1000 nM T25608 CV6O5J 127051856 EC50 = 187 nM T25608 CX7FO8 127051975 EC50 = 3690 nM T25608 CA0Z5S 127052270 EC50 = 1640 nM T25608 C9TX8Q 130253300 EC50 = 1200 nM T25608 CSI6R9 131842087 EC50 = 28.84 nM T25608 C1N5WO 131986027 EC50 = 13 nM T25608 C5IQ3Z 131986030 EC50 = 8 nM T25608 CB1ZH5 131986035 EC50 = 30 nM T25608 C47GLX 131986050 EC50 = 20 nM T25608 C7UQ4J 131986051 EC50 = 16 nM T25608 C5LZ8H 131986057 EC50 = 23 nM T25608 CYBU25 131986061 EC50 = 13 nM T25608 C8RL3X 131986065 EC50 = 88 nM T25608 CQW41S 131986072 EC50 = 15 nM T25608 C3HF5U 131986075 EC50 = 37 nM T25608 C4FK5N 131986082 EC50 = 67 nM T25608 CA5JX0 131986090 EC50 = 672 nM T25608 C4RI9P 131986112 EC50 = 54 nM T25608 C6WS3P 131986113 EC50 = 28 nM T25608 COCX92 131986115 EC50 = 18 nM T25608 CR13MG 131986116 EC50 = 12 nM T25608 CEZ01T 131986130 EC50 = 39 nM T25608 C6ZI8H 131986132 EC50 = 29 nM T25608 C0T6ZR 131986136 EC50 = 10 nM T25608 C6PY0T 131986140 EC50 = 19 nM T25608 C6FTO2 131986147 EC50 = 107 nM T25608 CQR4K9 131986162 EC50 = 858 nM T25608 C90AOL 131986164 EC50 = 134 nM T25608 CX91BM 131986179 EC50 = 15 nM T25608 CPGU02 131986182 EC50 = 85 nM T25608 C8W7DM 131986250 EC50 = 83 nM T25608 C3I8RE 131986294 EC50 = 9 nM T25608 C2RP7K 131986295 EC50 = 9 nM T25608 C4YV0A 131986297 EC50 = 63 nM T25608 C0L2GI 131986300 EC50 = 25 nM T25608 CF0XJ3 131986378 EC50 = 47 nM T25608 C9DIF2 131986401 EC50 = 20 nM T25608 CBXG19 132606863 EC50 = 110 nM T25608 C9IN6R 132606864 Ki = 45 nM T25608 CJ67MD 134129919 EC50 = 2.1 nM T25608 C53BMN 134129938 EC50 = 4400 nM T25608 CZBD80 134130352 EC50 = 58 nM T25608 CFH18E 134130696 EC50 = 61 nM T25608 CV7S3B 134130787 EC50 = 296 nM T25608 C0DU2R 134130822 EC50 = 1160 nM T25608 CHF3S7 134130859 EC50 = 1252 nM T25608 CSK3E0 134131511 EC50 = 7.3 nM T25608 C17CZB 134131620 EC50 > 10000 nM T25608 CW4S6G 134131874 EC50 > 10000 nM T25608 CO1RW6 134132142 EC50 > 9950 nM T25608 CXE17Y 134132711 IC50 > 100000 nM T25608 C4AB5J 134132951 EC50 > 10000 nM T25608 CB89WY 134133275 EC50 > 9950 nM T25608 C7DE1O 134133297 EC50 = 9260 nM T25608 CKTJ79 134133342 EC50 = 810 nM T25608 CG0L6Q 134133355 EC50 > 10000 nM T25608 CP92NR 134133506 EC50 > 20000 nM T25608 C2W0EY 134133675 EC50 = 3186 nM T25608 C83GOA 134133797 IC50 > 100000 nM T25608 CS3P7G 134133992 EC50 > 10000 nM T25608 CWS2G0 134134149 EC50 = 6799 nM T25608 CUEY64 134134226 EC50 > 20000 nM T25608 CJOQ95 134134229 EC50 = 1829 nM T25608 CQJ8M6 134134433 EC50 = 1.9 nM T25608 CK0NZ3 134134768 EC50 = 140 nM T25608 CNA4L8 134134846 IC50 = 173.78 nM T25608 C21VEN 134135255 EC50 > 20000 nM T25608 C96FRN 134135468 EC50 > 10000 nM T25608 CIFJ93 134135852 EC50 = 42 nM T25608 CUB2S6 134136015 EC50 = 1.4 nM T25608 CCH39I 134136175 EC50 = 6716 nM T25608 C1ECW4 134136203 EC50 = 38 nM T25608 CPBG95 134136959 EC50 = 280 nM T25608 C8LPH3 134137203 EC50 = 10 nM T25608 C2A1ZF 134137248 EC50 = 16.1 nM T25608 C7VOB4 134137619 EC50 > 9950 nM T25608 CR7P0U 134137873 EC50 = 10.5 nM T25608 CIRQ17 134137874 EC50 = 8.6 nM T25608 CXRE49 134138099 IC50 = 2884.03 nM T25608 CD9V6N 134138281 EC50 > 10000 nM T25608 CN9LG1 134138318 EC50 = 6311 nM T25608 CATP91 134138359 EC50 = 118.3 nM T25608 CF2RI3 134138706 EC50 = 16.7 nM T25608 C2J4UK 134138802 EC50 > 10000 nM T25608 C7K6EC 134138870 EC50 = 13 nM T25608 CBCK71 134139119 EC50 = 7 nM T25608 C5JM4L 134139171 EC50 = 2959 nM T25608 CPEK74 134139282 EC50 = 0.8 nM T25608 C1BMG7 134139527 EC50 = 2010 nM T25608 CTL96P 134139990 EC50 = 29.6 nM T25608 CGO7M3 134140070 EC50 > 10000 nM T25608 C5SQU0 134140073 EC50 > 9950 nM T25608 C8DM7J 134140466 EC50 = 2 nM T25608 C17WXH 134140675 EC50 = 4.4 nM T25608 C76URI 134141029 EC50 > 9950 nM T25608 CN9BG4 134141270 EC50 = 1126 nM T25608 CJ30RW 134141489 EC50 = 77 nM T25608 CI75ZW 134141650 IC50 = 3388.44 nM T25608 CO73WM 134141723 EC50 < 300 nM T25608 CNG6U9 134142024 EC50 > 20000 nM T25608 CAR2U0 134142025 EC50 > 20000 nM T25608 C35XWN 134142149 EC50 = 7.9 nM T25608 CZO53G 134142245 EC50 = 7.7 nM T25608 C6ZRV4 134142450 EC50 > 9950 nM T25608 CCDO98 134142866 EC50 = 4218 nM T25608 C4VL9A 134143163 EC50 > 9950 nM T25608 CIN93P 134143370 EC50 > 10000 nM T25608 C9LE7R 134143393 EC50 = 4540 nM T25608 C5HTX1 134143418 EC50 = 8.6 nM T25608 CBLF04 134143899 EC50 = 1391 nM T25608 C9QUR0 134144000 EC50 > 10000 nM T25608 CBW12L 134144214 EC50 = 9463 nM T25608 CL89UD 134144239 EC50 = 10 nM T25608 C0A8TH 134145071 IC50 > 100000 nM T25608 C2GH9K 134145195 EC50 > 9950 nM T25608 CYP7O1 134145412 EC50 > 9950 nM T25608 C8C1DB 134145700 EC50 > 10000 nM T25608 CU36BG 134145750 EC50 > 9950 nM T25608 C8KY5G 134145778 IC50 = 3890.45 nM T25608 C96FUD 134146021 EC50 > 9950 nM T25608 C9N5LO 134146386 EC50 > 10000 nM T25608 CY3ZF0 134146590 EC50 = 410 nM T25608 COYL20 134146720 EC50 > 10000 nM T25608 CC13ZE 134146958 EC50 > 10000 nM T25608 C1OMN0 134147174 EC50 > 9950 nM T25608 CXH3T0 134147328 IC50 = 19952.62 nM T25608 CJXK51 134147518 EC50 = 4.6 nM T25608 CUO72N 134147601 EC50 > 10000 nM T25608 CJ20TQ 134148110 EC50 > 10000 nM T25608 C6ZMV9 134148223 EC50 > 20000 nM T25608 C7XBW3 134148736 EC50 > 9950 nM T25608 CQ5R4P 134149615 EC50 = 1350 nM T25608 CA5B2J 134150245 EC50 = 1042 nM T25608 C9FZ5V 134150458 EC50 > 20000 nM T25608 C6Z7HO 134150797 EC50 = 1.9 nM T25608 C1GDK0 134150871 EC50 > 10000 nM T25608 C87ECV 134150969 EC50 > 1000 nM T25608 CLM9Q7 134151115 EC50 = 2504 nM T25608 CAG0Y1 134151150 EC50 = 55 nM T25608 CYG78X 134151354 EC50 > 20000 nM T25608 C6TP5Q 134151754 EC50 = 1270 nM T25608 CRH0A7 134151903 EC50 > 10000 nM T25608 CAY73T 134152336 EC50 > 10000 nM T25608 CF13KR 134152488 EC50 > 20000 nM T25608 C3SFX4 134152545 IC50 = 616.6 nM T25608 CNK25T 134152845 EC50 > 9950 nM T25608 CRGW59 134153067 IC50 = 44668.36 nM T25608 C82ZGH 134153148 EC50 = 71 nM T25608 CW54AS 134153222 IC50 > 100000 nM T25608 CVOE51 134153298 EC50 > 10000 nM T25608 C7U9SB 134153546 EC50 = 2000 nM T25608 C4H8UV 134153562 EC50 = 5406 nM T25608 C4O0ZM 134153986 EC50 > 10000 nM T25608 C49FKZ 134154330 EC50 > 9950 nM T25608 CV1E3G 134154415 EC50 > 10000 nM T25608 C0GYX7 134154417 EC50 > 9950 nM T25608 CM69QG 134154473 EC50 = 3600 nM T25608 C6SA1G 134154953 IC50 = 25118.86 nM T25608 CK29QG 134155067 EC50 > 10000 nM T25608 C9LNQ5 134155277 EC50 > 9950 nM T25608 CSM4R6 134155480 EC50 = 2100 nM T25608 CK7PY5 134155821 EC50 = 12 nM T25608 CA6RE0 134155847 EC50 = 2200 nM T25608 C7TO6A 134155950 EC50 > 10000 nM T25608 CK9M4A 134156096 EC50 = 3352 nM T25608 CL92ZI 134156455 EC50 > 10000 nM T25608 CA49BH 134156727 EC50 > 10000 nM T25608 CK84XB 134157015 EC50 = 1300 nM T25608 C7GDP1 134157207 EC50 > 9950 nM T25608 CJ6T8B 134157563 EC50 > 9950 nM T25608 C2GKN8 134157586 EC50 = 3586 nM T25608 CD0S5Z 134157824 EC50 > 20000 nM T25608 CUP4M1 134465730 EC50 = 2.2 nM T25608 CB0Q9N 134465732 EC50 = 0.2 nM T25608 C7V1RX 134465785 EC50 = 0.94 nM T25608 CVA5D0 134465794 EC50 = 0.25 nM T25608 CXOJ48 134538585 EC50 = 4 nM T25608 CKEP73 137529972 EC50 = 2 nM T25608 CRI0U6 137529979 EC50 = 148 nM T25608 CR4P2U 137529983 EC50 = 7 nM T25608 C8X1RQ 137631853 EC50 = 490 nM T25608 CYRS03 137632053 EC50 = 580 nM T25608 C7TA3H 137632403 EC50 > 30000 nM T25608 CBRG92 137633101 EC50 = 220 nM T25608 CUK0D4 137633394 EC50 = 150 nM T25608 C7MF0A 137633536 EC50 = 11800 nM T25608 CO0RD7 137633561 EC50 = 14800 nM T25608 C68SZA 137634330 EC50 = 81 nM T25608 CGE59Q 137634844 EC50 > 30000 nM T25608 CNUX64 137634863 EC50 > 33000 nM T25608 CL90AO 137634888 EC50 = 1260 nM T25608 C4JME8 137635143 EC50 = 2710 nM T25608 CCJ4W0 137635388 EC50 = 6400 nM T25608 C3IH5R 137635513 EC50 = 2320 nM T25608 CG8B5Y 137635715 EC50 = 260 nM T25608 COBJ62 137635907 EC50 = 70 nM T25608 COI40P 137636026 EC50 > 33000 nM T25608 CT0S7L 137636033 EC50 = 40100 nM T25608 CZ1OD2 137636167 EC50 = 1544 nM T25608 C6D7ZM 137636358 Ki = 49 nM T25608 C9GD8B 137636501 EC50 = 33500 nM T25608 CMO1E3 137636733 EC50 > 30000 nM T25608 C5QN8L 137637488 EC50 = 2100 nM T25608 CR53AY 137637576 EC50 = 3782 nM T25608 CL2DA0 137637602 EC50 = 1480 nM T25608 CWN80V 137638184 EC50 = 260 nM T25608 C3PO6D 137638269 EC50 = 220 nM T25608 CF35JS 137638341 EC50 = 180 nM T25608 CMPD78 137638355 EC50 = 18051 nM T25608 CE87QJ 137638413 EC50 = 1110 nM T25608 CT93OE 137638911 EC50 = 19952.62 nM T25608 CGD21L 137638995 EC50 = 7943.28 nM T25608 CR0IS1 137639817 EC50 = 450 nM T25608 CDMR25 137640032 EC50 = 6200 nM T25608 C0M8SI 137640301 EC50 = 1270 nM T25608 C4JOD5 137640323 EC50 > 30000 nM T25608 CI3R1P 137640417 EC50 = 32200 nM T25608 CUER14 137640728 EC50 = 3920 nM T25608 CP5U2V 137640781 EC50 = 900 nM T25608 CXL21U 137640919 EC50 = 680 nM T25608 CE9Z4L 137641343 EC50 = 19588 nM T25608 C4GVT6 137641734 EC50 = 13000 nM T25608 C0XLQ9 137642173 EC50 = 1210 nM T25608 CTW8I6 137642184 EC50 > 30000 nM T25608 CZ4KW8 137642604 EC50 = 7943.28 nM T25608 CNKP70 137642920 EC50 > 10000 nM T25608 C4QBG8 137642988 EC50 > 17000 nM T25608 CS59FT 137643339 EC50 = 10000 nM T25608 CJR49O 137643956 EC50 = 410 nM T25608 C1K4CL 137644843 EC50 = 82 nM T25608 CNK59T 137644989 EC50 = 110 nM T25608 C1XG9C 137645352 EC50 = 2560 nM T25608 CEYI29 137646043 EC50 = 11000 nM T25608 CM2C7J 137646188 EC50 > 30000 nM T25608 CU8OD6 137646308 EC50 = 640 nM T25608 CLTA84 137646337 EC50 = 6500 nM T25608 C19RYO 137646482 EC50 = 150 nM T25608 C7Y9PC 137646553 EC50 > 30000 nM T25608 C7SG5X 137646830 EC50 = 290 nM T25608 C4J7DH 137646898 EC50 > 33000 nM T25608 CIE72D 137647107 EC50 = 880 nM T25608 CQC17M 137647721 EC50 = 12589.25 nM T25608 C0OHT8 137648439 EC50 = 210 nM T25608 C3X4NA 137648780 EC50 = 240 nM T25608 C2DQ4O 137649008 Ki = 23000 nM T25608 CL1HE5 137649416 EC50 > 30000 nM T25608 CYX37M 137650524 EC50 = 2060 nM T25608 CCBI43 137652992 EC50 = 2420 nM T25608 CHD0E8 137653172 EC50 = 390 nM T25608 C9KHS5 137653756 EC50 = 3870 nM T25608 CBX4Z3 137653896 EC50 = 450 nM T25608 CFI68P 137653903 EC50 = 50 nM T25608 CP30FQ 137654021 EC50 = 210 nM T25608 CO2L0W 137654721 EC50 > 30000 nM T25608 C3Y9TQ 137655097 EC50 > 17000 nM T25608 C0XBY5 137655393 EC50 = 14700 nM T25608 CA3W9B 137655559 EC50 = 1140 nM T25608 CZLU59 137655619 EC50 = 1300 nM T25608 CT6S0B 137655758 EC50 > 33000 nM T25608 COB6K3 137656526 EC50 = 1423 nM T25608 C4E1YT 137657002 EC50 = 4600 nM T25608 CK5BX8 137657027 EC50 = 2010 nM T25608 CK9R6S 137657972 EC50 = 1584.89 nM T25608 CCW3P1 137658243 EC50 = 520 nM T25608 CCKT75 137658391 EC50 = 8900 nM T25608 CSR4W2 137658634 EC50 > 30000 nM T25608 C5YO8K 137658671 EC50 = 6490 nM T25608 CBG58K 137659266 EC50 = 260 nM T25608 CP96HY 137659517 EC50 = 680 nM T25608 CL70UQ 137659867 EC50 = 6100 nM T25608 CI21BK 137661056 EC50 = 2360 nM T25608 CT91BF 137661294 EC50 = 8 nM T25608 CZR62H 137661388 EC50 > 30000 nM T25608 CET37O 137661475 EC50 = 1700 nM T25608 CQ0GL8 137661929 EC50 = 57 nM T25608 C41OTE 141747238 EC50 = 4020 nM T25608 CDA4Z5 141747241 EC50 > 10000 nM T25608 C6K9ZT 142738539 EC50 = 9.4 nM T25608 CQ4TD1 142738540 EC50 > 25 nM T25608 CI71RX 142738543 EC50 = 1016 nM T25608 C02XYW 142738544 EC50 > 25 nM T25608 C08YVD 142738545 EC50 = 447 nM T25608 C60TYD 142738546 EC50 > 25 nM T25608 CO5ZN2 142738551 EC50 = 54.6 nM T25608 CAP4E3 142738553 EC50 = 778 nM T25608 CB7C3P 142738556 EC50 = 1308 nM T25608 CY6R9F 142738561 EC50 > 25 nM T25608 CI0E6S 142738567 EC50 = 37.8 nM T25608 C6I2JS 142738569 EC50 = 1800 nM T25608 C3R8IS 142738570 EC50 > 25 nM T25608 CCD2K8 142738574 EC50 > 25 nM T25608 CJ9B1F 142738575 EC50 = 1207 nM T25608 CBY8D4 142738578 EC50 > 25 nM T25608 C4LZ6A 142738583 EC50 = 1800 nM T25608 CQG5V4 145754982 EC50 = 41.69 nM T25608 CY0M8X 145949924 EC50 = 203 nM T25608 C74XZG 145949955 EC50 = 138 nM T25608 CN9KI4 145950126 EC50 = 172 nM T25608 C2L4ZC 145950191 EC50 = 531 nM T25608 CB7S9A 145950347 EC50 = 47 nM T25608 CYTD84 145950402 EC50 = 42 nM T25608 C8CZA1 145950447 EC50 = 54 nM T25608 CZQ1W4 145950728 EC50 = 113 nM T25608 C3UVA7 145951164 EC50 = 109 nM T25608 C0NML8 145951402 EC50 = 820 nM T25608 C09BIY 145952214 EC50 = 13 nM T25608 C6DOX5 145952673 EC50 = 50 nM T25608 CDLS51 145952700 EC50 = 1.6 nM T25608 CJ92XZ 145952952 EC50 = 20 nM T25608 CF1A8U 145953265 EC50 = 1136 nM T25608 CFP4H6 145953365 EC50 = 39 nM T25608 C7RGX9 145954367 EC50 = 94 nM T25608 C1S3NZ 145954394 EC50 > 10000 nM T25608 C6UT2R 145954794 EC50 = 155 nM T25608 CT2D7E 145954950 EC50 = 11330 nM T25608 CM3Y8D 145955179 EC50 = 308 nM T25608 CCP23Q 145955263 EC50 = 391 nM T25608 C4NM7D 145955723 EC50 = 231 nM T25608 C2O3LF 145955958 EC50 < 0.2 nM T25608 C9AJM4 145956000 EC50 > 1667 nM T25608 CLG81H 145956069 EC50 = 211 nM T25608 C2Q6IM 145956160 EC50 = 133 nM T25608 C1M5RN 145956406 EC50 < 0.2 nM T25608 C1GMP5 145956671 EC50 = 187 nM T25608 C0SLG1 145956739 EC50 = 610 nM T25608 CD6Y3Z 145956795 EC50 < 0.2 nM T25608 CLO4A7 145957072 EC50 = 97 nM T25608 CT7HW4 145957539 EC50 = 934 nM T25608 CR9J8V 145957609 EC50 = 1.1 nM T25608 CFD2Y6 145958651 EC50 > 10000 nM T25608 C36WRG 145958799 EC50 > 10000 nM T25608 C1IW4J 145958971 EC50 = 114 nM T25608 C1UB5H 145959273 EC50 = 8.2 nM T25608 CH6ZM0 145959598 EC50 = 57 nM T25608 CUG35K 145959722 EC50 = 417 nM T25608 CH8VA1 145959829 EC50 > 5000 nM T25608 CZ8E7J 145959985 EC50 = 1.7 nM T25608 CFGL96 145960084 EC50 = 1.6 nM T25608 C3A5XR 145960204 EC50 > 5000 nM T25608 CYHL49 145960453 EC50 = 21340 nM T25608 CV81UA 145960571 EC50 = 1.9 nM T25608 CMJ50D 145961418 EC50 = 0.8 nM T25608 CU14RO 145961656 EC50 = 5060 nM T25608 C9H0QO 145962064 EC50 = 144 nM T25608 CS8LJ9 145962072 EC50 = 179 nM T25608 CFUV91 145962164 EC50 = 4310 nM T25608 CD0W3C 145963128 EC50 > 25 nM T25608 C63OLJ 145963137 EC50 > 1667 nM T25608 CZ01IO 145963330 EC50 = 72 nM T25608 C9LH0Y 145963593 EC50 = 17750 nM T25608 CASW30 145963855 EC50 = 450 nM T25608 C9AQ6D 145964042 EC50 = 36.31 nM T25608 CS85LT 145964249 EC50 > 1000 nM T25608 CE09SL 145964735 EC50 > 10000 nM T25608 C6SHF7 145964802 EC50 = 426.58 nM T25608 CED62A 145964820 EC50 = 57.54 nM T25608 CH5MB9 145964866 EC50 > 1000 nM T25608 C1JR8C 145965138 EC50 = 257.04 nM T25608 C9SK7T 145965307 EC50 > 10000 nM T25608 CYT0J8 145965455 EC50 = 169.82 nM T25608 CPG7N1 145965467 EC50 = 331.13 nM T25608 CHZY25 145965661 EC50 = 52.48 nM T25608 CFX4L5 145965707 EC50 = 190.55 nM T25608 CJ1FL8 145965797 EC50 = 4120 nM T25608 CS9OA7 145965948 EC50 = 10500 nM T25608 C8RVW9 145965968 EC50 = 1411 nM T25608 CJK8U5 145965982 EC50 > 10000 nM T25608 CAL68F 145966017 EC50 = 1130 nM T25608 CE3BG0 145966029 EC50 > 10000 nM T25608 C74UGD 145966102 EC50 > 10000 nM T25608 C0L4YQ 145966167 EC50 = 457.09 nM T25608 C8R9YD 145966219 EC50 = 3260 nM T25608 C9D2XW 145966459 EC50 > 10000 nM T25608 C09WOF 145966485 EC50 = 1170 nM T25608 CG5QD9 145966540 EC50 > 1000 nM T25608 CU4GW5 145966632 EC50 = 251.19 nM T25608 C3IA4S 145966647 EC50 = 69.18 nM T25608 C2QT5B 145966699 EC50 = 213.8 nM T25608 C87MEW 145967080 EC50 > 10000 nM T25608 CNE6D4 145967091 EC50 = 66.07 nM T25608 CYC39X 145967263 EC50 = 177.83 nM T25608 CB57ZL 145967268 EC50 = 18600 nM T25608 CW6VO9 145967558 EC50 = 97.72 nM T25608 CU70AC 145967748 EC50 = 15.49 nM T25608 CX4BD7 145967778 EC50 = 75900 nM T25608 CCTO59 145967994 EC50 = 128.82 nM T25608 CIA03M 145968204 EC50 = 27.5 nM T25608 C7BTS4 145968322 EC50 = 157.1 nM T25608 C7FNC4 145969097 EC50 = 37.4 nM T25608 CR4BV2 145969373 EC50 > 10000 nM T25608 CKAL34 145969681 EC50 = 103.7 nM T25608 CMUN49 145970056 EC50 = 1020 nM T25608 CKRC96 145970067 EC50 > 1000 nM T25608 C0CVS9 145970371 EC50 = 53.7 nM T25608 CB6YO0 145970463 EC50 = 18.6 nM T25608 C7FY0C 145970728 EC50 = 28.9 nM T25608 CN4F0P 145971234 EC50 = 106 nM T25608 C1I9GA 145971547 EC50 > 10000 nM T25608 C7PCQ8 145971688 EC50 = 80 nM T25608 CIG73O 145971779 EC50 = 194.98 nM T25608 C9BZ7K 145971800 EC50 = 74.13 nM T25608 CW89VJ 145972020 EC50 = 133 nM T25608 CP0G4C 145972079 EC50 = 213.8 nM T25608 C3ZV6Y 145972304 EC50 = 1380 nM T25608 CWL07B 145973087 EC50 = 5020 nM T25608 C5ZTX4 145973102 EC50 > 10000 nM T25608 C12IJB 145973299 EC50 > 10000 nM T25608 C8X5FW 145973329 EC50 = 210 nM T25608 C2FN3Q 145973478 EC50 = 63.1 nM T25608 C96YWE 145973686 EC50 > 1000 nM T25608 C0CEN6 145973781 EC50 = 2540 nM T25608 CG28IX 145973933 EC50 > 10000 nM T25608 CAX4B9 145973937 EC50 = 1350 nM T25608 C13UBN 145973986 EC50 > 10000 nM T25608 C10LCU 145974034 EC50 > 1000 nM T25608 CQ8Z0G 145974173 EC50 = 170 nM T25608 C2NY0F 145974295 EC50 = 289 nM T25608 CI32AO 145974382 EC50 = 3670 nM T25608 CJUN-39 145974478 EC50 = 3090 nM T25608 CI50OB 145974495 EC50 = 46.77 nM T25608 CZV45O 145974509 EC50 = 2390 nM T25608 CQ9I5U 145974719 EC50 = 95.5 nM T25608 CL5TQ8 145975293 EC50 = 1520 nM T25608 C0B3CR 145975484 EC50 = 79.43 nM T25608 C0N4BC 145975522 EC50 = 5390 nM T25608 C2RPC5 145975621 EC50 = 2390 nM T25608 C4HRA6 145975628 EC50 = 288.4 nM T25608 CA21IS 145976136 EC50 = 275.42 nM T25608 CC52RT 145976145 EC50 = 194.98 nM T25608 CNL46D 145976172 EC50 = 234.42 nM T25608 C37RUC 145976267 EC50 = 1570 nM T25608 CGN2Y8 145976608 EC50 = 549.54 nM T25608 C07KYE 145976639 EC50 = 4 nM T25608 CD3R8O 145976702 EC50 = 2170 nM T25608 C2Z8KJ 145976748 EC50 = 234.42 nM T25608 CEP0I9 145976845 EC50 = 125.89 nM T25608 C59FXK 145976935 EC50 = 123.03 nM T25608 CHNC94 145976979 EC50 = 2430 nM T25608 CYI5W2 145977043 EC50 = 2710 nM T25608 C7TD1V 145977220 EC50 > 10000 nM T25608 CETA73 145977329 EC50 > 10000 nM T25608 CDTI80 145977404 EC50 = 269.15 nM T25608 C74JLM 145977668 EC50 = 363.08 nM T25608 CWA95F 145977707 EC50 = 1530 nM T25608 CS08HW 145977721 EC50 > 5000 nM T25608 CTM7A1 145977853 EC50 > 10000 nM T25608 C8MT3A 145978233 EC50 = 549.54 nM T25608 C6IU2A 145978511 EC50 = 51.29 nM T25608 C26HLU 145978559 EC50 > 1000 nM T25608 CXA80W 145978608 EC50 > 10000 nM T25608 CD67EV 145978633 EC50 = 7900 nM T25608 C0M4DC 145978849 EC50 > 1000 nM T25608 C9KC3V 145978975 EC50 = 3400 nM T25608 CLT09H 145979123 EC50 = 3980 nM T25608 C62KTQ 145979171 EC50 = 120 nM T25608 C5GLC7 145979252 EC50 = 4310 nM T25608 CC8E1Z 145979329 EC50 = 27200 nM T25608 C43IVG 145979602 EC50 = 36270 nM T25608 CXZ91W 145980154 EC50 = 10 nM T25608 CZ54IN 145980380 EC50 > 10000 nM T25608 CMUP96 145980455 EC50 = 13570 nM T25608 CN61AL 145980470 EC50 = 150 nM T25608 C0KP3F 145980573 EC50 = 3020 nM T25608 C1Q6PV 145980608 EC50 = 4260 nM T25608 CKR43C 145981599 EC50 = 3850 nM T25608 CPT0D9 145981771 EC50 = 830 nM T25608 C2SHF4 145981901 EC50 > 30000 nM T25608 CW9D3X 145981983 EC50 = 260 nM T25608 CUA9E3 145982071 EC50 = 980 nM T25608 CSW42Z 145982132 EC50 = 210 nM T25608 C87UAM 145982210 EC50 > 10000 nM T25608 CC2L9V 145982417 EC50 > 10000 nM T25608 CFY8U2 145982433 EC50 = 7620 nM T25608 C0JR7M 145982556 EC50 = 3000 nM T25608 CF34ZO 145982616 EC50 = 3500 nM T25608 CXY27B 145983006 EC50 = 61.5 nM T25608 CSW94B 145983457 EC50 = 5400 nM T25608 CO8K0Z 145983493 EC50 = 68780 nM T25608 C1CB9N 145983698 EC50 = 130 nM T25608 CAEZ16 145983824 EC50 = 3480 nM T25608 CS2A3B 145983825 EC50 = 76.4 nM T25608 CK9B5S 145984009 EC50 > 100000 nM T25608 C2IF8C 145984092 EC50 = 1200 nM T25608 C59PQC 145984275 EC50 = 800 nM T25608 C0OJ2P 145984445 EC50 > 100000 nM T25608 CT9V1W 145984594 EC50 > 100000 nM T25608 CKEB40 145984796 EC50 > 100000 nM T25608 C2V6CW 145984886 EC50 = 1030 nM T25608 CQ1TB7 145984906 EC50 = 3070 nM T25608 C67RHD 145984999 EC50 = 800 nM T25608 CK1IO9 145985116 EC50 = 2200 nM T25608 C0F2AH 145985122 EC50 = 11010 nM T25608 C9LV7A 145985123 EC50 = 93.7 nM T25608 C5C4YM 145985219 EC50 > 100000 nM T25608 CX4GB0 145985574 EC50 = 4000 nM T25608 C1HK7R 145985632 EC50 > 10000 nM T25608 CIGK40 145985686 EC50 = 24430 nM T25608 C5J4SE 145985748 EC50 > 100000 nM T25608 CX9U0T 145986046 EC50 = 29350 nM T25608 CPFW32 145986077 EC50 = 610 nM T25608 C28DAN 145986262 EC50 > 100000 nM T25608 CAE95K 145986458 EC50 > 10000 nM T25608 C0XPC2 145986478 EC50 > 50000 nM T25608 CDZG12 145986662 EC50 = 3060 nM T25608 CHL62X 145986689 EC50 = 8080 nM T25608 CW7Y4G 145986696 EC50 = 2380 nM T25608 CBOR53 145986704 EC50 > 10000 nM T25608 CT3W4M 145987015 EC50 = 100 nM T25608 C6DL2O 145987167 EC50 = 2870 nM T25608 C40HLG 145987309 EC50 = 5040 nM T25608 CB6QN4 145987484 EC50 = 7.9 nM T25608 C72DAS 145987796 EC50 = 200 nM T25608 C6MC4L 145987969 EC50 = 1800 nM T25608 CMN5R7 145987974 EC50 = 1470 nM T25608 CWZ5L7 145988414 EC50 = 39.7 nM T25608 C0G2WE 145988431 EC50 > 10000 nM T25608 CMBR98 145988551 EC50 > 10000 nM T25608 CTKM20 145988554 EC50 = 2850 nM T25608 C2ZBK5 145988796 EC50 = 210 nM T25608 CY2IL3 145989151 EC50 = 170 nM T25608 C75DSN 145989198 EC50 = 3590 nM T25608 CI94EP 145989566 EC50 = 2100 nM T25608 CHF9J1 145989900 EC50 = 2110 nM T25608 CI39OJ 145989913 EC50 > 10000 nM T25608 CQOK62 145990228 EC50 = 700 nM T25608 CJ76KD 145990303 EC50 = 2760 nM T25608 CT9WV6 145990337 EC50 = 8060 nM T25608 C7GK3H 145990715 EC50 = 46 nM T25608 C4BLV7 145990729 EC50 > 10000 nM T25608 C6OM1C 145990731 EC50 = 3770 nM T25608 CC28QH 145990980 EC50 = 110 nM T25608 C8CP3I 145991235 EC50 > 30000 nM T25608 CZQH15 145991380 EC50 = 5880 nM T25608 CVBP54 145991722 EC50 > 10000 nM T25608 CQ82EM 145991968 EC50 = 2370 nM T25608 CV2FB6 145992078 EC50 = 3450 nM T25608 C6F0LJ 145992170 EC50 = 3280 nM T25608 CP79UQ 145992176 EC50 > 10000 nM T25608 CEC30M 145992604 EC50 = 690 nM T25608 C0E2WQ 145992623 EC50 = 90 nM T25608 C87MWN 145992631 EC50 = 640 nM T25608 CDO7U1 145992642 EC50 = 2240 nM T25608 CCY19L 145992868 EC50 > 10000 nM T25608 CU3EG4 145993152 EC50 > 30000 nM T25608 CROV68 145993162 EC50 = 210 nM T25608 CX5FZ7 145993490 EC50 = 3870 nM T25608 C0T1BY 145993621 EC50 = 520 nM T25608 CFJQ16 145993644 EC50 = 280 nM T25608 C7DFI1 145994052 EC50 = 1170 nM T25608 CCV39B 145994196 EC50 = 8450 nM T25608 CC3SP5 146316684 EC50 = 6.1 nM T25608 C5BLX3 146695343 EC50 = 41.3 nM T25608 CG6T4L 146763588 EC50 = 59.8 nM T25608 CZGT59 146840871 EC50 = 40 nM T25608 C24OEI 147146439 EC50 = 4.8 nM T25608 CH2NL0 147329931 EC50 = 11.6 nM T25608 C0BDA4 147747458 EC50 = 38.7 nM T25608 C4G7NA 148173135 EC50 = 86.2 nM T25608 CIQ3X2 148485044 EC50 = 51.6 nM T25608 CP7I6Z 149144496 EC50 = 24.2 nM T25608 CDM45B 149231065 EC50 = 240 nM T25608 C1OK9A 149378333 EC50 = 225.3 nM T25608 CNWP21 149454889 EC50 = 19.3 nM T25608 CKH93B 153211729 EC50 = 196.7 nM T25608 CV53OY 153213696 EC50 = 58.5 nM T25608 C8LF3A 153272850 EC50 = 728.6 nM T25608 CM3H9E 155511380 EC50 = 220 nM T25608 C8Y9ST 155512244 EC50 = 374 nM T25608 C1N0VI 155512776 EC50 = 80 nM T25608 CYE8H1 155513821 EC50 = 59 nM T25608 C0VTM9 155515698 EC50 > 1000 nM T25608 C8RZH5 155515835 EC50 = 41.9 nM T25608 CM4TB2 155516498 EC50 = 54 nM T25608 CV53HO 155516879 EC50 = 120 nM T25608 CEZ0F1 155517179 EC50 = 1780 nM T25608 C08DTF 155517891 EC50 = 325 nM T25608 C93BFL 155519364 EC50 = 200 nM T25608 CU0L7Y 155522406 EC50 = 120 nM T25608 CT2H7E 155522452 EC50 = 460 nM T25608 C17OFD 155523655 EC50 = 1350 nM T25608 CPT9J8 155525700 EC50 = 185 nM T25608 C3P2ZK 155526024 EC50 > 10000 nM T25608 CAK2H8 155526126 EC50 = 220 nM T25608 C6RU2E 155526793 EC50 = 16 nM T25608 CWE06G 155527415 EC50 = 150 nM T25608 C26DHQ 155527487 EC50 = 60 nM T25608 CJP7Z9 155527626 EC50 = 326 nM T25608 CJI0N8 155527805 EC50 = 70 nM T25608 CR91BJ 155528372 EC50 = 2 nM T25608 C4SGK6 155528599 EC50 = 51.7 nM T25608 C34YXP 155529382 EC50 > 10000 nM T25608 CLV9W1 155529599 EC50 = 6500 nM T25608 C7NDX5 155529750 EC50 > 10000 nM T25608 C6N9YP 155530111 EC50 = 112 nM T25608 C69KEW 155530636 EC50 = 397.5 nM T25608 CT5D9K 155530726 EC50 > 10000 nM T25608 C41VZM 155533810 EC50 = 160 nM T25608 CBW2Z8 155535186 EC50 = 36.5 nM T25608 CVG6P0 155535946 EC50 > 10000 nM T25608 CXA3M2 155541840 EC50 = 536.2 nM T25608 CB14CD 155542122 EC50 = 80 nM T25608 C5W8SV 155543683 EC50 > 10000 nM T25608 CPU3Q0 155544661 EC50 = 11 nM T25608 C6PD1A 155545127 EC50 = 590 nM T25608 CX3KF2 155545207 EC50 > 10000 nM T25608 C1PO2Q 155546331 EC50 > 10000 nM T25608 CC63ZG 155547595 EC50 = 156 nM T25608 CR48CL 155547604 EC50 = 251 nM T25608 CEG6H0 155548030 EC50 = 400 nM T25608 CG3H7C 155548258 EC50 = 22.5 nM T25608 CZY63J 155549083 EC50 = 1.1 nM T25608 C9FV2A 155549085 EC50 = 36.1 nM T25608 CLI81V 155549391 EC50 = 1020 nM T25608 CAK8E6 155550483 EC50 = 45.6 nM T25608 C84OTS 155551422 EC50 = 0.11 nM T25608 CWHL51 155551584 EC50 = 16 nM T25608 CIK42F 155552554 EC50 = 290 nM T25608 CUAP95 155555299 EC50 > 10000 nM T25608 C4BSK6 155557354 EC50 > 10000 nM T25608 CY5RG0 155558174 EC50 = 69.6 nM T25608 CVH06N 155560437 EC50 > 10000 nM T25608 C7H1SI 155561223 EC50 = 155 nM T25608 CQ6VH4 155561358 EC50 = 247 nM T25608 C2NPT3 155561834 EC50 > 10000 nM T25608 C37ZFX 155563228 EC50 = 149 nM T25608 CQ7DF1 155565379 EC50 = 3 nM T25608 CG02XL 155565451 EC50 = 68 nM T25608 CS4UV7 155569570 EC50 = 300 nM T25608 C8H3WI 155569585 EC50 = 15.7 nM T25608 D01CCG 25150014 EC50 = 32 nM T25608 D01VIX 73777063 EC50 > 10000 nM T25608 D03JPL 79034 EC50 > 100000 nM T25608 D03LOG 5280450 EC50 = 540 nM T25608 D08MLH 46941175 Ki = 5.888 nM T25608 D08ZYC 11595431 EC50 = 13 nM T25608 D0C5SV 5280934 EC50 = 2884.03 nM T25608 D0J2EE 9957245 EC50 = 70 nM T25608 D0K6EG 57522038 EC50 = 5011.87 nM T25608 D0N0UC 3893 EC50 = 758.58 nM T25608 D0N9SV 25098573 EC50 = 9772.37 nM T25608 D0Q7BG 46854655 EC50 = 2.2 nM T25608 D0S0QY 66553168 EC50 = 5.888 nM T25608 D0T2CG 94216 EC50 > 100000 nM T25608 D0T4BP 97783 EC50 = 6760.83 nM T58741 D08HQK 5411 IC50 = 520 nM T58741 D0C7ET 11174599 IC50 = 2.3 nM T58741 D00BUR 216327 IC50 > 1000 nM T58741 D04PER 49836093 IC50 = 170 nM T58741 D0K9IF 71666749 IC50 > 30000 nM T58741 D0O7QA 46840946 IC50 = 160 nM T58741 D0OX9F 16046068 IC50 = 15000 nM T58741 CPN25U 998021 IC50 = 10300 nM T58741 CZK6M0 22239024 IC50 = 660 nM T58741 C3LK1F 42637004 IC50 = 1030 nM T58741 C40BIM 45139151 IC50 = 1050 nM T58741 CS5EJ1 46841648 IC50 = 1636 nM T58741 CRE97F 46841787 IC50 = 1109 nM T58741 C06OXV 52920492 IC50 = 24000 nM T58741 CMS2F7 53239561 IC50 = 3320 nM T58741 CC82DM 65459349 IC50 = 4200 nM T58741 C2MC6B 71522734 IC50 = 0.8 nM T58741 CM1B0W 71523649 IC50 = 46000 nM T58741 CJXK67 71559365 IC50 = 11 nM T58741 C9MUK3 71716856 IC50 = 510 nM T58741 CUG2V3 71716866 IC50 = 199 nM T58741 C15BSO 86270136 IC50 = 190 nM T58741 CTG76E 86687532 IC50 = 3700 nM T58741 C1BIF8 90026208 IC50 = 38 nM T58741 C26BZK 91666633 IC50 = 92 nM T58741 C7NLE8 91809347 IC50 = 480 nM T58741 CC5N9I 117737142 IC50 = 1300 nM T58741 C10BKY 117749324 IC50 = 650 nM T58741 C9KV7L 117993993 IC50 = 9400 nM T58741 C7AYV5 118540795 IC50 = 5.461 nM T58741 CR8TX9 118708662 IC50 = 26 nM T58741 C9JL4Y 118937760 IC50 = 8600 nM T58741 C9Q2ND 121333973 IC50 = 16000 nM T58741 C9K5RV 122513516 IC50 > 20000 nM T58741 C09QIY 127047645 IC50 = 5000 nM T58741 CF6L8Q 145955101 IC50 = 66 nM T58741 CCTB54 145958837 IC50 = 104 nM T58741 C38DYW 145959291 IC50 = 183 nM T58741 CK7PN3 145969142 IC50 = 1600 nM T58741 C8Q2EG 145988110 IC50 = 2100 nM T58741 COZ54G 155523716 IC50 = 1000 nM T58741 C5F9BQ 155526497 IC50 = 29000 nM T58741 CE3H4Z 155567528 IC50 = 130 nM T58741 D0P8TL 56947150 IC50 = 1.1 nM T04696 D0W0VD 3885 IC50 = 970 nM T04696 CW68ZS 61672 IC50 = 40000000 nM T04696 CH67EZ 91286 IC50 = 4100 nM T04696 CZTD26 220436 IC50 = 9000 nM T04696 CVGN02 267570 IC50 > 30000 nM T04696 CE7M6K 269624 IC50 = 40 nM T04696 CRSF26 304992 IC50 > 111000 nM T04696 CSO78Y 322478 EC50 = 870 nM T04696 CZ34CV 349435 IC50 = 25000 nM T04696 CS2B8E 397888 IC50 = 1000 nM T04696 C9WI3X 460748 EC50 = 780 nM T04696 CWYT28 460749 EC50 = 430 nM T04696 CIJ28W 555805 IC50 > 111000 nM T04696 C4BRI2 707946 IC50 > 100000 nM T04696 C6WZ2C 866938 EC50 > 30000 nM T04696 C7WC0L 930115 EC50 > 30000 nM T04696 CJ0V3O 931081 EC50 > 30000 nM T04696 CK1TD5 941846 EC50 > 30000 nM T04696 C0ME8D 951230 EC50 = 7360 nM T04696 CB0X4T 951368 EC50 > 30000 nM T04696 CBN32K 1293987 IC50 > 100000 nM T04696 C6LPN3 1313201 IC50 > 100000 nM T04696 CRL05A 1771058 IC50 = 32000 nM T04696 C35DCU 3164059 EC50 = 510 nM T04696 CNTJ89 3164066 EC50 = 1070 nM T04696 CSXC46 3164070 EC50 = 330 nM T04696 C2C9RE 4989139 EC50 = 300 nM T04696 CO01XP 5478021 IC50 = 3500 nM T04696 CO8M4Q 6411132 EC50 > 20000 nM T04696 C2BY6K 6458554 EC50 = 960 nM T04696 CVC31J 6459022 EC50 = 290 nM T04696 CC6U7A 6493950 EC50 = 280 nM T04696 C5FY6T 11266171 IC50 = 7600 nM T04696 C65MLO 11840607 IC50 = 23600 nM T04696 CHDB52 12023317 IC50 = 11000 nM T04696 C1JX2C 12023323 IC50 = 3500 nM T04696 C4RGJ6 14895314 IC50 > 111000 nM T04696 C54WZY 14895315 IC50 = 43000 nM T04696 C8Z9XB 16481078 EC50 = 200 nM T04696 CK7J6D 17756791 EC50 = 3500 nM T04696 CFBT48 46833159 EC50 = 680 nM T04696 COS86H 46834048 EC50 = 750 nM T04696 CV60DR 46834317 EC50 = 370 nM T04696 CCM26J 56837840 IC50 > 111000 nM T04696 C0DMZ7 57400600 IC50 > 111000 nM T04696 CS0Q9C 59299967 IC50 = 19000 nM T04696 CZ3Y7S 60103948 IC50 > 111000 nM T04696 CWJ46V 60104019 IC50 > 111000 nM T04696 C5BJM9 68699178 IC50 > 111000 nM T04696 CU8ZA0 71817697 EC50 = 260 nM T04696 CLD4B7 71817698 EC50 = 400 nM T04696 CZE8Q2 71817849 EC50 = 4630 nM T04696 CG2A6C 71817850 EC50 = 280 nM T04696 C2ZYW4 71817852 EC50 > 10000 nM T04696 C35QBR 71817853 EC50 = 7420 nM T04696 C8A0CS 71818002 EC50 = 670 nM T04696 CHKS75 71818003 EC50 = 1020 nM T04696 CJ3YG9 71818004 EC50 = 700 nM T04696 C8WN0H 71818005 EC50 = 640 nM T04696 C4HGP6 71818006 EC50 = 430 nM T04696 CEX8A6 71818007 EC50 = 150 nM T04696 CPB21Q 71818143 EC50 = 770 nM T04696 CTD4U6 71818144 EC50 = 250 nM T04696 C7UB6O 71818145 EC50 = 120 nM T04696 CHF45Y 71818146 EC50 = 50 nM T04696 C96AYZ 71818147 EC50 > 20000 nM T04696 CJ2OV6 71818149 EC50 > 20000 nM T04696 CLAF94 71818291 EC50 = 2100 nM T04696 CWHG19 71818293 EC50 > 150000 nM T04696 CH6BV1 71818296 EC50 > 150000 nM T04696 CHN47D 71818443 EC50 > 150000 nM T04696 CZXW74 71818444 EC50 > 150000 nM T04696 CTSD96 71818445 EC50 > 30000 nM T04696 C2WO0L 71818446 EC50 > 30000 nM T04696 C1Z9HD 71818447 EC50 > 30000 nM T04696 CG7Q6D 71818587 EC50 > 30000 nM T04696 CW8N0J 71818588 EC50 > 30000 nM T04696 C3M4FP 71818589 EC50 > 30000 nM T04696 C69KUV 71818590 EC50 > 30000 nM T04696 CT30QA 71818591 EC50 > 30000 nM T04696 C3WJ6B 71818592 EC50 > 30000 nM T04696 C7TIJ1 71818716 EC50 > 30000 nM T04696 CLU15O 71818717 EC50 > 30000 nM T04696 CF9I3P 71818718 EC50 > 30000 nM T04696 C3DTB4 71818719 EC50 > 30000 nM T04696 CI80ND 71818720 EC50 > 30000 nM T04696 COU9C7 71818721 EC50 > 30000 nM T04696 C8AR0I 71818722 EC50 = 1660 nM T04696 CB23IX 71818723 EC50 > 30000 nM T04696 CQV2B5 71818864 EC50 = 480 nM T04696 C8L1XF 71818865 IC50 = 27480 nM T04696 C5CXH0 71818866 EC50 = 2870 nM T04696 C7P2XN 71818867 EC50 = 500 nM T04696 CPK26T 71818868 IC50 = 42 nM T04696 C85OTM 71818869 EC50 = 90 nM T04696 CK6W2Z 71818870 EC50 = 250 nM T04696 C9MKT5 71819004 EC50 = 470 nM T04696 CMI5O8 71819005 EC50 = 1040 nM T04696 CG7ZN2 71819006 EC50 = 320 nM T04696 CWSE58 71819007 EC50 = 3390 nM T04696 CXG20Y 71819008 EC50 = 2740 nM T04696 CMT0Y2 71819009 EC50 = 90 nM T04696 C48DOI 71819143 EC50 = 30 nM T04696 CJC48A 71819144 EC50 = 4660 nM T04696 C7GXZ3 71819145 EC50 = 1370 nM T04696 C7Q0NF 71819146 EC50 = 290 nM T04696 C5ET9H 71819147 EC50 = 640 nM T04696 CRZ8G6 71819148 EC50 = 370 nM T04696 C19SNE 71819283 IC50 = 41 nM T04696 CB4NR9 72211790 IC50 = 9800 nM T04696 C6NQP9 73346151 EC50 = 720 nM T04696 C9CI3X 73350770 EC50 = 360 nM T04696 CRZ62F 73355036 EC50 = 24000 nM T04696 CSP7U6 118641028 IC50 > 111000 nM T04696 COJ93Q 121472570 IC50 = 11000 nM T04696 CE8KX5 121472571 IC50 = 35000 nM T04696 CU2O3F 121478289 IC50 = 11000 nM T04696 CJ1E0R 121478290 IC50 = 12000 nM T04696 C2UMF7 121478292 IC50 > 111000 nM T04696 C0SM2F 121478293 IC50 = 51000 nM T04696 C41BGD 121478294 IC50 = 15000 nM T04696 C3V9CO 121478295 IC50 = 16000 nM T04696 C7R5DK 121478296 IC50 = 66000 nM T04696 C7FYP6 121478298 IC50 > 111000 nM T04696 CIRH72 121478299 IC50 > 111000 nM T04696 CG9MA0 121478300 IC50 = 7700 nM T04696 C2NCD1 121478303 IC50 = 13000 nM T04696 CQ71GI 121478304 IC50 > 111000 nM T04696 C2JEM3 121478305 IC50 = 3300 nM T04696 CV37KR 121478306 IC50 > 111000 nM T04696 CHZ3G9 121478307 IC50 = 11000 nM T04696 C6LQR0 121478308 IC50 = 12000 nM T04696 CY52IG 121478317 IC50 = 50000 nM T04696 CD7O9U 121478318 IC50 = 24000 nM T04696 CB46CR 121478319 IC50 = 13000 nM T04696 CWN68V 121478326 IC50 = 13000 nM T04696 C5QRF9 121478327 IC50 = 14000 nM T04696 C2LGQ0 121478328 IC50 = 17000 nM T04696 COSM56 121478329 IC50 = 13000 nM T04696 CAI2T3 121478330 IC50 = 10000 nM T04696 C2UHT5 121478331 IC50 = 10000 nM T04696 C3QXM6 121478332 IC50 > 111000 nM T04696 C4GFH8 121478333 IC50 = 12000 nM T04696 CG48YT 121478334 IC50 = 8100 nM T04696 C3YM8C 121478345 IC50 = 19000 nM T04696 CUH40X 121478347 IC50 = 17000 nM T04696 CDY7B5 121478349 IC50 > 111000 nM T04696 C0P8VG 121478351 IC50 = 1900 nM T04696 CKC14X 121478358 IC50 = 37000 nM T04696 C0G9RA 121478361 IC50 = 14000 nM T04696 C27CJU 121478363 IC50 = 71000 nM T04696 CH30JX 121478365 IC50 = 22000 nM T04696 CQ3CR2 121478367 IC50 = 19000 nM T04696 CW12NY 121478368 IC50 = 68000 nM T04696 CN9UE4 121478394 IC50 = 9800 nM T04696 CCW7Y0 121478397 IC50 = 13000 nM T04696 C9B2OZ 121478399 IC50 = 11000 nM T04696 C5CN6W 121478400 IC50 = 8800 nM T04696 C1WC5X 121478401 IC50 = 18000 nM T04696 C9M1LP 121478402 IC50 = 6600 nM T04696 CN5QF3 121478403 IC50 > 111000 nM T04696 CI53LJ 121478405 IC50 = 24000 nM T04696 C12FTJ 121478406 IC50 > 111000 nM T04696 CJLG39 121478407 IC50 = 12000 nM T04696 C60YRK 121478438 IC50 > 111000 nM T04696 CT1RL3 122179149 IC50 > 111000 nM T04696 CM9AU7 122179162 IC50 > 111000 nM T04696 C98KOJ 122179163 IC50 = 37000 nM T04696 C7Q9FC 122179164 IC50 > 111000 nM T04696 CTFO36 122483585 IC50 = 5500 nM T04696 C2Q1HV 122483587 IC50 = 6500 nM T04696 CVE37N 122483588 IC50 = 13000 nM T04696 CSCZ94 122483589 IC50 = 18000 nM T04696 CU8C3T 122483590 IC50 = 7100 nM T04696 C9X8QL 122483591 IC50 = 30000 nM T04696 CM20BN 122483592 IC50 = 2600 nM T04696 COC53H 122483593 IC50 = 3200 nM T04696 CE89RT 122483594 IC50 > 37000 nM T04696 C15GNW 122483596 IC50 > 37000 nM T04696 CUGI76 122483597 IC50 = 10000 nM T04696 CCLF45 122483598 IC50 = 4500 nM T04696 CH9OJ3 122483599 IC50 > 111000 nM T04696 CIPC52 122483600 IC50 = 26000 nM T04696 C04XUJ 122483601 IC50 = 14000 nM T04696 CG3O5N 122483604 IC50 = 25000 nM T04696 C6W8SH 122483605 IC50 > 37000 nM T04696 CSOF59 122483606 IC50 = 16000 nM T04696 C4QH5Y 122483608 IC50 = 9300 nM T04696 C6FZQ4 122483609 IC50 = 16000 nM T04696 C7Q3LI 122483610 IC50 = 5200 nM T04696 C1WCV3 122483611 IC50 > 111000 nM T04696 C5UVQ3 122483612 IC50 = 3300 nM T04696 CN1W3U 122483613 IC50 > 111000 nM T04696 C2EX1V 122483614 IC50 = 4100 nM T04696 C4PG1R 122483615 IC50 = 4500 nM T04696 C52AQF 122483618 IC50 > 111000 nM T04696 CNO57Z 122483619 IC50 = 16000 nM T04696 CH95QN 122483620 IC50 = 36000 nM T04696 C9B0TV 122483622 IC50 = 42000 nM T04696 CV7H2F 122483623 IC50 > 111000 nM T04696 C5X8OF 122483624 IC50 = 3000 nM T04696 C8Q6ZY 122483625 IC50 = 4500 nM T04696 CSKF94 122483626 IC50 = 1900 nM T04696 CG6U2L 122483627 IC50 = 20000 nM T04696 CGB0R9 122483628 IC50 = 19000 nM T04696 C41LDF 122483629 IC50 = 21000 nM T04696 C8MC5T 122483630 IC50 = 25000 nM T04696 C8C9SW 122483631 IC50 = 5400 nM T04696 CW0KF2 122483633 IC50 = 14000 nM T04696 CAST90 122483634 IC50 = 23000 nM T04696 C0DBQ9 122483635 IC50 = 2700 nM T04696 CRDV43 122483636 IC50 = 50000 nM T04696 C2DEL7 122483637 IC50 = 11000 nM T04696 C3KDP2 122483638 IC50 = 11000 nM T04696 CGZ75H 122483639 IC50 = 11000 nM T04696 CP87QX 122483641 IC50 = 15000 nM T04696 C7BL9T 122484905 IC50 = 6300 nM T04696 C3FS6Y 122484906 IC50 = 8900 nM T04696 CT5OG6 127028881 IC50 = 5100 nM T04696 CPY24W 127029757 IC50 > 111000 nM T04696 C7YX4G 127030613 IC50 > 111000 nM T04696 CLT35C 127043728 IC50 > 111000 nM T04696 CJA2I1 127044083 IC50 = 37000 nM T04696 CBFS34 127044239 IC50 > 111000 nM T04696 CE15TB 127044402 IC50 > 111000 nM T04696 CF64IU 127044403 IC50 > 111000 nM T04696 C12IUQ 127044404 IC50 > 111000 nM T04696 CBE49O 127044405 IC50 > 111000 nM T04696 CM19WU 127044406 IC50 = 111000 nM T04696 CU15SD 127044408 IC50 = 111000 nM T04696 C0X5YU 127044409 IC50 = 111000 nM T04696 C3XO0J 127044411 IC50 > 111000 nM T04696 COX07F 127044412 IC50 > 111000 nM T04696 C5OQ3T 127044413 IC50 > 111000 nM T04696 C38YZG 127044414 IC50 > 111000 nM T04696 C0SP4E 127044557 IC50 > 111000 nM T04696 CPEU65 127044559 IC50 > 111000 nM T04696 C1W8YR 127044560 IC50 > 111000 nM T04696 CPWI81 127051466 IC50 = 12000 nM T04696 C9L1GO 129896914 IC50 = 12000 nM T04696 C5DA0Z 135163962 IC50 = 37000 nM T04696 C3OGL8 135438987 IC50 = 17700 nM T04696 C5K9YU 136236292 IC50 = 17000 nM T04696 CQZ79S 137633472 IC50 > 111000 nM T04696 CEMW84 137634763 IC50 = 1000 nM T04696 CY83RB 137635101 IC50 = 61600 nM T04696 CY4BH7 137635982 IC50 = 12000 nM T04696 CP8I0N 137635992 IC50 = 107000 nM T04696 CC1X7N 137637372 IC50 > 111000 nM T04696 CSKE17 137638583 IC50 > 111000 nM T04696 C7K5XB 137638718 IC50 > 111000 nM T04696 CY0G2M 137639745 IC50 = 32900 nM T04696 CE93VQ 137639878 IC50 = 108000 nM T04696 C7KVT8 137640123 IC50 = 37000 nM T04696 C7EHL1 137643195 IC50 > 111000 nM T04696 CQ89WF 137644721 IC50 > 111000 nM T04696 C7LY3U 137645346 IC50 > 111000 nM T04696 CT8A6V 137645479 IC50 = 37000 nM T04696 CTD0Q1 137645708 IC50 = 37000 nM T04696 C83FEH 137646143 IC50 > 111000 nM T04696 CR72BP 137646560 IC50 = 37000 nM T04696 CW24CA 137650951 IC50 > 111000 nM T04696 C2RVW9 137651075 IC50 > 111000 nM T04696 C7SUD6 137652086 IC50 = 104000 nM T04696 C9X2IG 137652438 IC50 > 111000 nM T04696 CY25WR 137653301 IC50 > 111000 nM T04696 CDQ41E 137656446 IC50 > 111000 nM T04696 CZ01OK 137658578 IC50 = 37000 nM T04696 CHXA46 137659333 IC50 = 37000 nM T04696 CB9GY3 137660083 IC50 > 111000 nM T04696 C09XQR 137661166 IC50 > 111000 nM T04696 CSB6M0 139368816 IC50 = 130 nM T04696 C84UBZ 139368818 IC50 = 65 nM T04696 CQ4G6B 139368820 IC50 = 70 nM T04696 C3F9GV 139368834 IC50 = 6.5 nM T04696 CWL01S 139368851 IC50 = 3800 nM T04696 CQ0F4V 139368854 IC50 = 320 nM T04696 CBM15W 139368874 IC50 = 20 nM T04696 CNI9A6 139368879 IC50 = 14 nM T04696 C5M1BA 139368887 IC50 = 880 nM T04696 CEH93B 139368894 IC50 = 33 nM T04696 CBM19D 139368902 IC50 = 7.3 nM T04696 CE9AK7 139368907 IC50 = 930 nM T04696 CQD73C 139368913 IC50 = 38 nM T04696 CS9UM7 139368918 IC50 = 200 nM T04696 CD9HM5 139368920 IC50 = 35 nM T04696 C2PUL4 139368923 IC50 = 300 nM T04696 CPDJ72 139368930 IC50 = 1100 nM T04696 C5G7JZ 139368935 IC50 = 6.1 nM T04696 C0AM4H 139368936 IC50 = 270 nM T04696 CVF8C5 139368940 IC50 > 10000 nM T04696 C8VH9F 139368954 IC50 = 190 nM T04696 CBI70J 139368955 IC50 = 150 nM T04696 CDW39J 139368964 IC50 = 33 nM T04696 C30ENM 139368966 IC50 = 960 nM T04696 CMP03R 139368970 IC50 = 1600 nM T04696 CT95OC 139368975 IC50 = 1500 nM T04696 C7EH0V 139368985 IC50 = 1000 nM T04696 C1LBE4 139368987 IC50 = 380 nM T04696 CC3QT9 139379823 IC50 = 990 nM T04696 C5Y2ZA 145949905 IC50 > 111000 nM T04696 CUL1I3 145950046 IC50 = 99000 nM T04696 CF6Y7J 145950454 IC50 > 111000 nM T04696 CDM0W7 145951675 IC50 = 28000 nM T04696 CEO83W 145952632 IC50 = 36000 nM T04696 C47WUP 145952847 IC50 > 111000 nM T04696 C74VYG 145953711 IC50 = 51000 nM T04696 CV35UN 145954864 IC50 = 24000 nM T04696 C0WC6Q 145955087 IC50 > 111000 nM T04696 CZ54YB 145955773 IC50 = 88000 nM T04696 C9IPA5 145956858 IC50 = 31000 nM T04696 C4UTW8 145957109 IC50 > 111000 nM T04696 CRA1K8 145957662 IC50 = 12000 nM T04696 C5X9ZY 145957721 IC50 = 38000 nM T04696 C1QE7V 145958498 IC50 = 29000 nM T04696 C3CHN5 145958644 IC50 = 28000 nM T04696 CUYA76 145959663 IC50 > 111000 nM T04696 C4NU9M 145960096 IC50 > 111000 nM T04696 C2X5SP 145972895 IC50 > 111000 nM T04696 C3DCY1 145973141 IC50 = 31000 nM T04696 C93HRO 148522856 IC50 = 1300 nM T04696 CUFI09 155511226 IC50 = 22000 nM T04696 C1OUY2 155511648 IC50 = 77300 nM T04696 CXY2T9 155513626 IC50 > 100000 nM T04696 CR06GW 155516031 IC50 > 100000 nM T04696 C82ZWB 155517851 IC50 = 80900 nM T04696 CSQ6J0 155520530 IC50 > 100000 nM T04696 C1UFN8 155520960 IC50 > 100000 nM T04696 C1F8SC 155521790 IC50 > 100000 nM T04696 CRQ5V4 155522028 IC50 > 100000 nM T04696 C2TAG8 155522368 IC50 > 100000 nM T04696 CYT67S 155522639 IC50 > 100000 nM T04696 CJ2YD3 155523314 IC50 = 80800 nM T04696 CKI09P 155527507 IC50 > 100000 nM T04696 C7GYW1 155527618 IC50 > 100000 nM T04696 CE1KY2 155527688 IC50 > 100000 nM T04696 CB4WA6 155527846 IC50 > 100000 nM T04696 CN4XT5 155528962 IC50 > 100000 nM T04696 CMS31Q 155529562 IC50 > 100000 nM T04696 C5CK8O 155530724 IC50 > 100000 nM T04696 CE6SN1 155532734 IC50 > 100000 nM T04696 C3FKI7 155533180 IC50 > 100000 nM T04696 C1BYP0 155534526 IC50 > 100000 nM T04696 CT81JB 155536721 IC50 > 100000 nM T04696 CTD2N5 155537102 IC50 = 43800 nM T04696 C9PV4T 155537144 IC50 = 85200 nM T04696 CU13XE 155539442 IC50 > 100000 nM T04696 C6V8HO 155541099 IC50 = 21000 nM T04696 CV1YX3 155546559 IC50 > 100000 nM T04696 C9J0VW 155547447 IC50 > 100000 nM T04696 C5BL8C 155547740 IC50 > 100000 nM T04696 C8OH9M 155548958 IC50 > 100000 nM T04696 C3DO8S 155550002 IC50 > 100000 nM T04696 CVM59F 155550044 IC50 > 100000 nM T04696 C01UYS 155553494 IC50 > 100000 nM T04696 C5ZR0U 155553817 IC50 > 100000 nM T04696 C4MT7Q 155561437 IC50 > 100000 nM T04696 C3A2VZ 155563144 IC50 = 94500 nM T04696 CI36HO 155563834 IC50 = 59000 nM T04696 CR0IP2 155564579 IC50 > 100000 nM T04696 CZ6R9X 155565688 IC50 > 100000 nM T04696 CXEY68 155566971 IC50 > 100000 nM T04696 C5EG2O 155567730 IC50 = 16600 nM T04696 CYHT71 155568211 IC50 > 100000 nM T04696 C0ST7X 155568568 IC50 > 100000 nM T04696 D0J1KH 262093 IC50 = 71000 nM T04696 D0P0CM 460747 EC50 = 1160 nM T16633 D0TV0C 9941444 Ki = 6.31 nM T16633 D06JFI 11251755 IC50 = 27 nM T16633 D0J8PI 158782 IC50 > 10000 nM T16633 D0L9QM 59568713 IC50 = 2630 nM T16633 D09JXL 5311430 Ki < 1000 nM T16633 C6XYL5 6918011 Ki = 501.19 nM T16633 CHM63P 6918026 Ki = 158.49 nM T16633 CR0U6E 9827283 Ki = 5382 nM T16633 CA8UQ7 9848232 Ki = 4264 nM T16633 CTRI07 9852911 Ki = 4000 nM T16633 C9BJ3Q 9854636 IC50 > 1000 nM T16633 CDU75Z 9857566 Ki = 5000 nM T16633 CMLP16 9918828 Ki = 630.96 nM T16633 C3Z5YJ 9963342 Ki = 3.981 nM T16633 CIT57N 9985523 Ki = 4100 nM T16633 C64LIB 10009650 Ki = 300 nM T16633 CL6G0Z 10094509 Ki = 2310 nM T16633 C9C7RK 10096510 Ki = 9700 nM T16633 CFZN71 10166743 Ki = 1730 nM T16633 CI21CK 10179247 Ki > 10000 nM T16633 C6DRE9 10210016 Ki = 1550 nM T16633 C4M9GN 10248767 Ki = 3400 nM T16633 C78LUH 10296743 Ki = 1400 nM T16633 CSY5K2 10325243 Ki = 2400 nM T16633 CL87OB 10411795 Ki = 2600 nM T16633 CS96ON 10534086 IC50 = 1000 nM T16633 CHZ9I8 10554930 Ki = 6800 nM T16633 CY3ZE9 10577746 IC50 = 501 nM T16633 C9C0HF 10580397 Ki = 2100 nM T16633 CU3DQ6 10630127 Ki = 1000 nM T16633 C45JIZ 10699714 Ki = 4400 nM T16633 CG2UX4 10701257 IC50 = 1000 nM T16633 CP0F7C 10724811 IC50 = 1000 nM T16633 C3TMY5 10724880 IC50 = 1580 nM T16633 CJM47E 10748701 IC50 = 2163 nM T16633 CWF2N5 10748831 IC50 = 1000 nM T16633 CLW4V6 10770814 Ki = 4000 nM T16633 CO56HI 10772403 IC50 = 1000 nM T16633 CGN0Z5 10772578 IC50 = 535 nM T16633 C3L4DH 10796238 IC50 = 4843 nM T16633 C15QGO 10819673 IC50 = 1000 nM T16633 CFL71O 10843862 IC50 = 1000 nM T16633 C2PJ1O 10876898 Ki = 10 nM T16633 C6TVQ8 10964197 Ki = 6.31 nM T16633 CXDG12 10996788 Ki = 1.585 nM T16633 C6AW0M 11112736 Ki > 10000 nM T16633 CK1RX4 11136828 Ki = 63.1 nM T16633 CR1JP9 11147505 Ki = 3.981 nM T16633 C1I9EX 11159133 IC50 = 757 nM T16633 C7REL4 11170698 IC50 = 117 nM T16633 CIEM12 11170867 IC50 > 10000 nM T16633 CW2JA8 11182381 IC50 = 410 nM T16633 CE3GC2 11205475 IC50 = 5.3 nM T16633 CXI32T 11205496 IC50 = 450 nM T16633 C2RNJ5 11205515 IC50 = 327 nM T16633 CUT8Z0 11240205 IC50 = 21 nM T16633 CK78SD 11240206 IC50 = 27 nM T16633 C67WXD 11274767 IC50 = 10.3 nM T16633 COK06N 11320738 IC50 > 1000 nM T16633 C5D6AM 11332138 IC50 > 1000 nM T16633 C5PAN4 11343811 IC50 > 1000 nM T16633 CLQ53A 11355270 IC50 = 410 nM T16633 CQ0UC7 11378229 IC50 = 607 nM T16633 CC09ZU 11378299 IC50 > 1000 nM T16633 CG7PT9 11389178 IC50 = 650 nM T16633 CFJD72 11423410 IC50 = 330 nM T16633 C4S2HG 11434734 IC50 = 49 nM T16633 C6XHC3 11457491 IC50 = 213 nM T16633 CJ5A9B 11457521 IC50 = 840 nM T16633 CMA8C7 11468709 IC50 > 10000 nM T16633 CG8A0J 11468887 IC50 = 6.5 nM T16633 CZ3N5J 11468916 IC50 = 55 nM T16633 CORY59 11480246 IC50 = 545 nM T16633 C63QMX 11535351 IC50 > 1000 nM T16633 CF6K7M 11563877 IC50 = 5100 nM T16633 CS68YA 11642413 IC50 = 9590 nM T16633 CZHN61 11678313 IC50 > 10000 nM T16633 CW65KY 11705763 Ki = 530 nM T16633 CN63YV 11787877 IC50 > 10000 nM T16633 CR6UF9 11788180 IC50 > 1000 nM T16633 CK4U8N 11804376 IC50 = 1000 nM T16633 C9XH7F 11815114 Ki = 1.585 nM T16633 CRA01O 11845058 IC50 > 1000 nM T16633 C8X3CL 11845059 IC50 > 1000 nM T16633 CO3HT9 11847587 IC50 > 1000 nM T16633 CMR10F 11848679 Ki = 1750 nM T16633 CBV2X0 11963995 Ki = 5100 nM T16633 CW7I8U 13690207 Ki = 224 nM T16633 C8OU7I 15429504 IC50 = 723 nM T16633 CEO3F0 15585102 IC50 > 1000 nM T16633 CC2YJ8 16062553 Ki > 10000 nM T16633 C3H1RT 16062555 Ki > 10000 nM T16633 C1LH5T 16062816 Ki = 4500 nM T16633 C1GKF8 16130982 Ki = 0.32 nM T16633 C2TRA5 16144717 IC50 = 1044 nM T16633 CW20OC 16144977 IC50 = 506 nM T16633 CS6A3Z 16145268 IC50 = 1000 nM T16633 CN3LS1 16145579 IC50 = 1000 nM T16633 C72MUC 16146425 IC50 = 1000 nM T16633 CD91IL 16148220 IC50 = 1000 nM T16633 C59OUC 16148481 Ki = 125.89 nM T16633 CJG1X9 16148596 Ki = 0.631 nM T16633 CNY09C 16148922 Ki = 1000 nM T16633 CP0DC8 16149640 Ki = 0.5012 nM T16633 CDPC19 16149975 Ki = 6.31 nM T16633 C0SE6V 16150676 Ki = 0.2512 nM T16633 CSP6A9 16150915 Ki = 0.1585 nM T16633 C6N7SR 16151159 Ki = 19.95 nM T16633 C2B9IL 16151570 IC50 = 189 nM T16633 CQM8J1 16151781 IC50 = 347 nM T16633 CM8UF7 16151826 IC50 = 3.3 nM T16633 CJ7UT6 16151923 IC50 > 1000 nM T16633 CIM03U 16152257 IC50 = 270 nM T16633 CU7X6V 16153077 IC50 = 88 nM T16633 CK4O1V 16153193 IC50 = 517 nM T16633 C16LMW 16153418 IC50 > 1000 nM T16633 CO0LG7 16154000 IC50 = 99 nM T16633 CX4RM8 16154096 IC50 = 13 nM T16633 COYU86 16156815 Ki = 1000 nM T16633 CI3FW1 16157160 IC50 = 1025 nM T16633 C7GN0S 16157479 Ki = 0.1995 nM T16633 CQL5O0 16181427 IC50 = 31 nM T16633 C2CUY9 16181428 EC50 = 33 nM T16633 CUH8D7 16737812 IC50 > 1000 nM T16633 C8QIT3 16737813 IC50 > 1000 nM T16633 CNP36U 16737814 IC50 = 233 nM T16633 C7Q6JL 16738359 IC50 = 89 nM T16633 C6F1RZ 24777672 IC50 = 961 nM T16633 C5GZO7 24858018 IC50 = 96 nM T16633 CV1U7H 24858920 IC50 = 14 nM T16633 C0UB7K 24859055 IC50 > 1000 nM T16633 CQCW58 24859056 IC50 = 22 nM T16633 CT6J2A 24859195 IC50 = 16 nM T16633 CUDV69 24859196 IC50 > 1000 nM T16633 C45NYA 24859341 IC50 > 1000 nM T16633 C4AB6I 24859342 IC50 = 416 nM T16633 CH50QU 24859494 IC50 = 79 nM T16633 C8L2KJ 24859495 IC50 > 1000 nM T16633 CDS6W5 24859645 IC50 = 358 nM T16633 CHF20D 24859646 IC50 > 1000 nM T16633 CKH2R4 24859787 IC50 = 540 nM T16633 CT1BM6 24859788 IC50 > 1000 nM T16633 C2IKX3 24859919 IC50 > 1000 nM T16633 C5OQ2X 24859920 IC50 > 1000 nM T16633 CSZ73L 24860057 IC50 > 1000 nM T16633 C36ZHQ 24860058 IC50 > 1000 nM T16633 CVL48C 24860201 IC50 = 302 nM T16633 C20ZFS 24860202 IC50 = 218 nM T16633 CHKC79 25187396 IC50 = 253 nM T16633 C4YXJ1 25187398 IC50 = 54 nM T16633 CO9PI7 25187400 IC50 = 27 nM T16633 C8C9PL 25187679 IC50 = 38 nM T16633 C9ECD8 25187681 IC50 > 1000 nM T16633 C43OES 25187683 IC50 = 247 nM T16633 CNTB73 25187685 IC50 = 89 nM T16633 C1IUQ2 25187953 IC50 = 837 nM T16633 CQ3F8L 25187955 IC50 = 379 nM T16633 CS2ZV1 25188218 IC50 = 630 nM T16633 CLI2U1 25188220 IC50 = 183 nM T16633 CNDU95 25188496 IC50 = 962 nM T16633 C7KF8N 25188776 IC50 > 1000 nM T16633 CCHN50 25188780 IC50 = 105 nM T16633 C3T8DA 25189052 IC50 = 76 nM T16633 CI21ED 25189054 IC50 = 372 nM T16633 C97LHK 25189325 IC50 = 75 nM T16633 CEG4J0 25189327 IC50 = 387 nM T16633 CSQH26 42637069 EC50 = 3.9 nM T16633 CJ1S9K 42637136 IC50 = 37 nM T16633 C3NYM8 42637137 IC50 = 97 nM T16633 CJ47CL 42637210 IC50 = 530 nM T16633 CR3A8Q 42637283 IC50 = 189 nM T16633 CENZ47 42637363 IC50 = 108 nM T16633 CX0JC7 42637503 IC50 = 0.19 nM T16633 C90LHS 42637563 IC50 = 4.7 nM T16633 C80WBK 42637632 IC50 = 8.2 nM T16633 CR49YE 42637984 IC50 > 1000 nM T16633 CEFO24 42638065 IC50 = 150 nM T16633 CF5JK4 42638066 IC50 = 14 nM T16633 CHY04A 44290718 IC50 > 1000 nM T16633 C16BKW 44290734 IC50 > 1000 nM T16633 CW76YB 44290735 IC50 > 1000 nM T16633 CA6IS7 44290766 IC50 > 1000 nM T16633 C6BZ1J 44298104 Ki = 348 nM T16633 CCXL10 44298113 Ki > 1000 nM T16633 CYW8O0 44298130 Ki = 1690 nM T16633 CB9JK1 44298131 Ki = 1030 nM T16633 CJ5WL8 44298155 Ki > 1000 nM T16633 CHL57J 44298156 Ki = 1200 nM T16633 CP61LB 44298165 Ki > 1000 nM T16633 CM0B6J 44298166 Ki > 1000 nM T16633 C8XZR7 44298169 Ki = 1060 nM T16633 C0DPX7 44298171 Ki = 413 nM T16633 C62OEU 44298177 Ki = 82 nM T16633 CS9JW8 44298178 Ki > 1000 nM T16633 C20MBI 44298179 Ki = 1950 nM T16633 C3QBP0 44298188 Ki = 525 nM T16633 C1R3QD 44298189 Ki = 575 nM T16633 C5RJ7U 44298195 Ki = 435 nM T16633 C8N3EJ 44298197 Ki = 443 nM T16633 CZU05A 44298214 Ki > 1000 nM T16633 CQUS98 44298218 Ki = 37 nM T16633 COTK07 44298219 Ki = 186 nM T16633 CAJO07 44298231 Ki = 415 nM T16633 C9S4IX 44298232 Ki = 845 nM T16633 CB1A3K 44298235 Ki = 174 nM T16633 C2TQ1V 44298248 Ki = 69 nM T16633 C3WFV5 44298250 Ki = 374 nM T16633 CVW19Y 44298328 Ki = 34 nM T16633 CT94HY 44298329 Ki = 568 nM T16633 CL4F1V 44298378 Ki = 238 nM T16633 CMO1Q9 44298441 Ki = 1400 nM T16633 C8Y9ZP 44298443 Ki > 1000 nM T16633 CUSR45 44298468 Ki > 1000 nM T16633 C8EN2H 44298469 Ki = 60 nM T16633 CWE7Q0 44298482 IC50 = 245 nM T16633 CF69PL 44298522 Ki = 484 nM T16633 CRQJ98 44308836 Ki = 537 nM T16633 CRFM02 44308969 Ki = 1.6 nM T16633 C40MJU 44308970 Ki = 0.38 nM T16633 C9KR7Q 44309052 Ki = 2430 nM T16633 C4YG1S 44311590 IC50 = 30.9 nM T16633 CY0OV9 44311591 IC50 = 309 nM T16633 C29GQB 44311601 IC50 = 1 nM T16633 CC8DS0 44311602 IC50 = 450 nM T16633 C5KST2 44311690 IC50 = 35 nM T16633 C6N4MH 44311691 IC50 = 530 nM T16633 CIR4G6 44311695 IC50 = 17.4 nM T16633 CTG6X5 44311696 IC50 = 2.5 nM T16633 C7Y8SF 44311697 IC50 = 8.1 nM T16633 CK52MY 44311702 IC50 = 15.1 nM T16633 CX39CV 44311703 IC50 = 187 nM T16633 C5RM2A 44311730 IC50 = 15 nM T16633 CBG70T 44311731 IC50 = 24 nM T16633 CQH20F 44311765 IC50 > 1000 nM T16633 CZG4K6 44311836 IC50 = 33 nM T16633 CWNP79 44311837 IC50 = 34.7 nM T16633 CWSF38 44311868 IC50 = 103 nM T16633 C2T0YP 44311869 IC50 = 101 nM T16633 C1ONB3 44311870 IC50 = 347 nM T16633 C1GY0F 44311912 IC50 = 3.6 nM T16633 C14DIH 44311913 IC50 > 1000 nM T16633 C1X4TI 44311914 IC50 = 27.3 nM T16633 C64WAE 44311958 IC50 = 130 nM T16633 CFT90E 44311959 IC50 > 1000 nM T16633 C3PQD0 44311960 IC50 = 720 nM T16633 CS7PB4 44312258 IC50 > 1000 nM T16633 C5PE1D 44325273 IC50 = 407 nM T16633 C1P0QV 44332931 Ki = 1800 nM T16633 CHP41F 44363816 Ki = 712 nM T16633 CH2DN4 44367916 IC50 > 10000 nM T16633 CM9YQ0 44367953 IC50 > 10000 nM T16633 C5W4YL 44368019 IC50 = 667 nM T16633 CO6ZJ9 44368020 IC50 > 1000 nM T16633 CQ5T1D 44368043 IC50 > 1000 nM T16633 C1SWO5 44368044 IC50 > 10000 nM T16633 C29EZK 44368080 IC50 = 778 nM T16633 C9ZW6U 44368093 IC50 > 1000 nM T16633 C71URM 44368094 IC50 > 1000 nM T16633 CC1ZP9 44368109 IC50 > 10000 nM T16633 CQ7OP1 44368112 IC50 > 1000 nM T16633 C0EW4I 44368117 IC50 > 1000 nM T16633 C6TNZ9 44368144 IC50 > 1000 nM T16633 C53IAG 44368153 IC50 = 545 nM T16633 CKU8J7 44368156 IC50 = 5.3 nM T16633 CR12GB 44368157 IC50 = 27 nM T16633 C50DMO 44368226 IC50 > 10000 nM T16633 CN31HS 44368398 IC50 > 1000 nM T16633 C2RC0P 44368406 IC50 = 45 nM T16633 CB1HC8 44368422 IC50 > 10000 nM T16633 C27DLY 44368489 IC50 > 10000 nM T16633 CWHK38 44377332 Ki > 10000 nM T16633 CVH1O7 44377366 Ki > 5000 nM T16633 CRC2N1 44377555 Ki = 2900 nM T16633 CS1WT5 44377591 Ki = 4000 nM T16633 C3LUY8 44377623 Ki > 10000 nM T16633 CQD0P4 44377645 Ki > 5000 nM T16633 CWNF42 44385504 Ki = 2570 nM T16633 CAFD79 44385508 Ki > 10000 nM T16633 CHY14B 44385591 Ki = 9100 nM T16633 CJQI19 44385652 Ki = 1520 nM T16633 CG12HD 44385712 Ki = 2840 nM T16633 C8MU5C 44385757 Ki = 1880 nM T16633 C0LRT9 44386389 Ki = 3430 nM T16633 C1EVK8 44387399 Ki = 1030 nM T16633 C6U9VC 44388027 IC50 = 14 nM T16633 C2IW5J 44388028 IC50 = 6.1 nM T16633 C27ANT 44388029 IC50 = 46 nM T16633 CHQK20 44388035 IC50 > 1000 nM T16633 CI9XS1 44388036 IC50 = 259 nM T16633 CD4BX6 44388037 IC50 = 620 nM T16633 CDS08Z 44388038 IC50 > 1000 nM T16633 CZA03Y 44388040 IC50 > 1000 nM T16633 C21WBR 44388043 IC50 > 1000 nM T16633 C7VK6B 44388052 IC50 > 1000 nM T16633 CT93BI 44388060 IC50 = 597 nM T16633 C4E5VS 44388061 IC50 > 1000 nM T16633 C7P5RO 44388066 IC50 > 1000 nM T16633 C7T8IY 44388069 IC50 = 208 nM T16633 C2TWO3 44388070 IC50 > 1000 nM T16633 CDBE87 44388075 IC50 = 5.2 nM T16633 C25GWK 44388078 IC50 > 1000 nM T16633 CT93LV 44388079 IC50 > 1000 nM T16633 CX54SC 44388083 IC50 = 53 nM T16633 C2C0RU 44388084 IC50 = 144 nM T16633 C5SMA2 44388085 IC50 = 255 nM T16633 C26OCG 44388086 IC50 = 30 nM T16633 C8SR2O 44388087 IC50 = 35 nM T16633 CHL5T1 44388088 IC50 > 1000 nM T16633 C4VNC2 44388089 IC50 > 1000 nM T16633 C1IH3T 44388090 IC50 > 1000 nM T16633 CNC91I 44388093 IC50 = 5.8 nM T16633 CN45OF 44388095 IC50 = 8.5 nM T16633 C82HJL 44388104 IC50 = 241 nM T16633 CV6T2H 44388105 IC50 = 554 nM T16633 CLC0N2 44388106 IC50 = 53 nM T16633 C0VO1K 44388107 IC50 = 94 nM T16633 CM5O3B 44388108 IC50 = 16 nM T16633 CAF02P 44388109 IC50 = 782 nM T16633 C23XBM 44388110 IC50 = 204 nM T16633 CPX74G 44388112 IC50 = 22 nM T16633 CG9SA3 44388114 IC50 = 43 nM T16633 C2C4MH 44388116 IC50 = 17 nM T16633 CW1EL5 44388118 IC50 > 1000 nM T16633 CN0K3V 44388119 IC50 = 74 nM T16633 CE8DH4 44388120 IC50 = 61 nM T16633 C1A0OY 44388121 IC50 = 3.3 nM T16633 CS53NP 44388122 IC50 > 1000 nM T16633 CX67WG 44388123 IC50 = 6.7 nM T16633 CB50EK 44388124 IC50 = 4.8 nM T16633 C9SN1X 44388132 IC50 = 64 nM T16633 C6W4YT 44388133 IC50 = 167 nM T16633 CMTN20 44388134 IC50 = 274 nM T16633 CAK42W 44388135 IC50 = 89 nM T16633 CTW48B 44388136 IC50 = 181 nM T16633 C4P1AS 44388137 IC50 = 18 nM T16633 CEAZ82 44388138 IC50 = 62 nM T16633 C1KMT8 44397389 Ki = 58 nM T16633 CN6Z8C 44397648 Ki = 180 nM T16633 CRW0M6 44397706 Ki = 130 nM T16633 CM1R8X 44400000 IC50 > 10000 nM T16633 CP89CS 44400135 IC50 > 10000 nM T16633 C1BY2P 44444935 IC50 > 1000 nM T16633 CH17TI 44560858 IC50 > 1000 nM T16633 C2AZY7 44560859 IC50 > 1000 nM T16633 C2I8NB 44560860 IC50 > 1000 nM T16633 C4XRT0 44560861 IC50 > 1000 nM T16633 C21TZI 44560862 IC50 > 1000 nM T16633 C2YM5N 44560863 IC50 > 1000 nM T16633 CS39FB 44560864 IC50 > 1000 nM T16633 CU3FD2 44560865 IC50 > 1000 nM T16633 C8IKU1 44560866 IC50 > 1000 nM T16633 CTQ83Z 44560867 IC50 > 1000 nM T16633 CQC29N 44560868 IC50 > 1000 nM T16633 C47MDA 44560869 IC50 > 1000 nM T16633 CHAJ41 44560870 IC50 > 1000 nM T16633 CT0A9U 44560871 IC50 > 1000 nM T16633 CM0T9R 44560872 IC50 > 1000 nM T16633 CO2J6R 44560873 IC50 > 1000 nM T16633 CKQD64 44560874 IC50 > 1000 nM T16633 CEK26Y 44560875 IC50 > 1000 nM T16633 CBL1P7 44560876 IC50 > 1000 nM T16633 CY47DM 44560877 IC50 > 1000 nM T16633 C5OZD1 44560878 IC50 > 1000 nM T16633 CFT47C 44560898 IC50 > 1000 nM T16633 CAO7R0 44560899 IC50 > 1000 nM T16633 C80ZCF 44560900 IC50 > 1000 nM T16633 CATH94 44560901 IC50 > 1000 nM T16633 C2AXG6 44560902 IC50 > 1000 nM T16633 COQ9W7 44560903 IC50 > 1000 nM T16633 CLZ23V 44560904 IC50 > 1000 nM T16633 C0OKG2 44560905 IC50 > 1000 nM T16633 CPIW17 44560906 IC50 > 1000 nM T16633 CFR3Y5 44560907 IC50 > 1000 nM T16633 CS85LR 44560908 IC50 > 1000 nM T16633 C6K1FI 44577218 IC50 > 1000 nM T16633 CAJ15T 44577219 IC50 > 1000 nM T16633 CQD56E 44577220 IC50 > 1000 nM T16633 CV18IC 44577221 IC50 = 763 nM T16633 CLJD09 45102042 IC50 > 10000 nM T16633 C63YJS 45139239 IC50 > 1000 nM T16633 C63XPN 45267999 IC50 > 1000 nM T16633 CF09UA 45268875 IC50 = 1 nM T16633 CU3MQ4 45268876 EC50 = 0.93 nM T16633 C2PNH4 45272264 IC50 = 17 nM T16633 CFL9K7 45273129 IC50 > 1000 nM T16633 C9Z4MR 45273130 IC50 > 1000 nM T16633 C4RGN0 45273131 IC50 = 20 nM T16633 C6KBJ2 46882133 Ki = 4950 nM T16633 CU1D6I 46902023 IC50 = 2800 nM T16633 CZ46AH 46911015 IC50 < 300 nM T16633 C84ZTC 49865341 IC50 > 1000 nM T16633 C3VZ4U 49865342 IC50 > 1000 nM T16633 CGYR09 49865343 IC50 = 25 nM T16633 C35WID 49865344 IC50 > 1000 nM T16633 C0RK7G 49865345 IC50 = 1000 nM T16633 C4YLM7 49865346 IC50 > 1000 nM T16633 CZ4RI1 49865347 IC50 = 57.5 nM T16633 C9SNL1 52941607 IC50 > 10000 nM T16633 C40ZRY 52948630 IC50 > 10000 nM T16633 CED3O6 53473658 IC50 = 138 nM T16633 CE7J0U 53473659 IC50 = 140 nM T16633 CY0G2K 53473744 IC50 = 2.7 nM T16633 CBQG96 53473824 IC50 = 4.1 nM T16633 CW53YV 53473917 IC50 > 1000 nM T16633 C87SME 53474004 IC50 > 1000 nM T16633 C7EO1Z 53474005 IC50 > 1000 nM T16633 CY3M2A 53474090 IC50 > 1000 nM T16633 C9JHI4 56664813 Ki = 2 nM T16633 C8ZW3O 56927659 IC50 = 2362 nM T16633 CHK8T1 56945132 Ki = 4750 nM T16633 C73XBL 57384077 IC50 > 1000 nM T16633 C3KC9Z 57398462 IC50 = 3.2 nM T16633 C0DEM2 68254010 IC50 = 6000 nM T16633 CTVI05 70683416 IC50 = 267 nM T16633 CV42WQ 70689221 IC50 > 10000 nM T16633 C3P0AN 70689413 IC50 > 1000 nM T16633 CP58HL 70689414 IC50 > 1000 nM T16633 CB14OW 70689415 IC50 > 1000 nM T16633 CNZC97 70689723 IC50 = 1.2 nM T16633 C2WQM9 70691295 IC50 > 1000 nM T16633 C5E8MY 70693613 IC50 > 1000 nM T16633 C3TZ9U 70695246 IC50 = 495 nM T16633 C34XGS 70695722 IC50 > 1000 nM T16633 CIPF50 70695723 IC50 > 1000 nM T16633 CF08XL 71458043 Ki = 4600 nM T16633 CU82HG 71460000 IC50 = 975 nM T16633 CPC69G 71461645 Ki = 3300 nM T16633 CLAV92 71461684 IC50 > 1000 nM T16633 C1NZU3 71461685 IC50 = 563 nM T16633 CFKH42 71717904 IC50 = 2003 nM T16633 CGDO59 72947672 Ki = 0.31 nM T16633 CIO28F 73345407 Ki = 1000 nM T16633 CMN6X8 73345525 IC50 > 10000 nM T16633 C70XZC 73345528 IC50 > 1000 nM T16633 CXGJ67 73345700 IC50 > 1000 nM T16633 CV23JS 73345701 IC50 > 1000 nM T16633 C81UME 73345740 Ki > 1000 nM T16633 CX5VM1 73346900 IC50 = 443 nM T16633 CA3MU5 73346903 IC50 = 5.4 nM T16633 C62NFY 73346927 Ki = 1000 nM T16633 CK64MX 73346930 Ki = 1000 nM T16633 C15CAN 73346972 Ki > 1000 nM T16633 CD09FU 73347225 Ki > 1000 nM T16633 CI4L6W 73347226 Ki = 736 nM T16633 CGM61R 73348311 Ki > 10000 nM T16633 CN1FD2 73348312 Ki = 4400 nM T16633 C01GIQ 73348427 Ki = 1000 nM T16633 C7Y9ZT 73348428 Ki = 1000 nM T16633 CFLT50 73348719 IC50 > 1000 nM T16633 C75NBQ 73348741 Ki > 1000 nM T16633 C5MNX3 73348742 Ki > 1000 nM T16633 CL94MY 73350006 Ki = 1000 nM T16633 C0N6XK 73350010 Ki = 1000 nM T16633 CTV30F 73350011 Ki = 1000 nM T16633 CF2AK4 73350012 Ki = 1000 nM T16633 CK9CS4 73351516 Ki = 1000 nM T16633 CNY13O 73351517 Ki = 1000 nM T16633 CUN6L1 73351622 IC50 = 607 nM T16633 CC98JE 73351624 IC50 > 1000 nM T16633 CWUH52 73351718 Ki = 1000 nM T16633 CS9I4W 73351829 Ki > 1000 nM T16633 CF70XH 73351873 IC50 = 104 nM T16633 CFB54J 73352985 Ki = 1395 nM T16633 CKFV85 73353009 Ki > 1000 nM T16633 CC45AV 73353272 IC50 > 10000 nM T16633 C41OCY 73353278 IC50 > 1000 nM T16633 CW54CU 73353340 IC50 > 1000 nM T16633 CL7DT2 73354494 Ki = 1000 nM T16633 CA48EL 73354535 Ki > 1000 nM T16633 CFK7Z3 73354633 IC50 > 10000 nM T16633 C1UYL2 73354783 IC50 > 1000 nM T16633 CG1CX0 73354798 IC50 > 1000 nM T16633 CIVZ67 73354818 Ki > 1000 nM T16633 CGCE64 73354819 Ki > 1000 nM T16633 C1Y0CI 73356066 Ki = 1000 nM T16633 C52JAS 73356068 Ki = 395 nM T16633 CN5LG8 73356069 Ki = 1000 nM T16633 C9GKV2 73356181 IC50 = 323 nM T16633 C7XFB6 73356331 IC50 > 1000 nM T16633 CI02SE 73356366 Ki > 1000 nM T16633 CW8L6C 76310862 IC50 > 1000 nM T16633 CHV6K7 76314485 IC50 = 18 nM T16633 C0PR3Y 76314486 IC50 > 1000 nM T16633 C94BWD 76314487 IC50 = 38 nM T16633 C25XKO 76314488 IC50 = 171 nM T16633 CS54IV 76321777 IC50 = 33 nM T16633 C94OAT 76321778 IC50 = 795 nM T16633 CU1IR8 76325402 IC50 = 14 nM T16633 CL09JQ 86279005 IC50 > 10000 nM T16633 C3JOS4 86292350 Ki > 9090 nM T16633 CVLE34 86293506 Ki = 848 nM T16633 C15VTO 86294248 Ki = 4535 nM T16633 C2BAV8 90644981 Ki = 656 nM T16633 CI58FM 90663867 IC50 > 1000 nM T16633 CK62FO 90663868 IC50 > 10000 nM T16633 C7AFD4 90663869 IC50 > 1000 nM T16633 C94XTF 90663872 IC50 > 10000 nM T16633 CA7W0U 90663873 IC50 > 10000 nM T16633 C4EG8T 90663874 IC50 > 10000 nM T16633 CW21UO 90663875 IC50 > 1000 nM T16633 C7Q4PD 90665458 Ki = 153000 nM T16633 CR43ZL 90665459 Ki = 102000 nM T16633 CLK7C3 90665460 Ki = 16000 nM T16633 CZ0UC6 90665461 Ki = 8200 nM T16633 C0IBJ6 90665462 Ki = 16000 nM T16633 CPX0C9 90665463 Ki = 12000 nM T16633 C3UVC8 91936728 IC50 > 10000 nM T16633 CT3UP7 91936729 IC50 > 10000 nM T16633 CD2E4L 101941290 IC50 = 1000 nM T16633 C9KB3W 117711399 Ki = 7360 nM T16633 CTH52C 118718416 Ki = 0.7943 nM T16633 CKQ4P6 118718462 IC50 = 945 nM T16633 C1Z7UJ 118718463 Ki < 1000 nM T16633 CPYA80 118718465 IC50 = 1000 nM T16633 CR61UD 118718466 IC50 = 1000 nM T16633 CW64XN 118718500 IC50 = 1000 nM T16633 CB4D5T 118718501 IC50 = 3219 nM T16633 CW5HG2 118718502 IC50 = 1000 nM T16633 CC36KP 118718503 IC50 = 1086 nM T16633 C7FIQ1 118718504 IC50 = 1008 nM T16633 CNBY57 118718505 IC50 = 1000 nM T16633 CPY4Q5 118718506 IC50 = 245 nM T16633 CO13JR 118718507 IC50 = 1000 nM T16633 CLFJ60 118718508 IC50 = 1439 nM T16633 C13YUH 118718509 IC50 = 588 nM T16633 CP2O7U 118718510 IC50 = 1000 nM T16633 CLDZ63 118718511 IC50 = 1000 nM T16633 CYQ7X2 118718854 IC50 > 1000 nM T16633 CA6C4T 118719101 IC50 = 397 nM T16633 CDZ3H4 118719196 IC50 > 1000 nM T16633 CQRO32 118719197 IC50 > 1000 nM T16633 CGXH91 118719198 IC50 > 1000 nM T16633 C1QJX7 118719199 IC50 > 1000 nM T16633 C0GLC8 118719200 IC50 > 10000 nM T16633 C40NGQ 118719201 IC50 > 10000 nM T16633 CK2W9T 118719202 IC50 > 1000 nM T16633 CW4AT0 118719275 IC50 > 10000 nM T16633 C5VWI1 118719303 IC50 = 1665 nM T16633 CS12JW 122179457 IC50 = 2300 nM T16633 CNGQ19 122179477 IC50 = 1330 nM T16633 CE79SV 138377584 IC50 > 10000 nM T16633 CE76TG 42637005 IC50 = 591 nM T16633 C6ELN4 42637006 IC50 = 356 nM T16633 CS73LG 42637433 IC50 = 449 nM T16633 C6C3YF 45270549 IC50 = 2.5 nM T16633 C9Y3BS 45270550 IC50 = 6.1 nM T16633 CQC51Z 45270552 IC50 > 1000 nM T16633 CXE30U 45271377 IC50 = 3.6 nM T16633 D01BWV 9802572 Ki = 3700 nM T16633 D01NID 44388055 IC50 = 71 nM T16633 D02CQW 11847438 IC50 > 1000 nM T16633 D02NJV 44388048 IC50 = 189 nM T16633 D02OJQ 44388115 IC50 = 10 nM T16633 D02WOX 44388129 IC50 = 33 nM T16633 D03DRL 44388045 IC50 = 176 nM T16633 D03SXC 44388041 IC50 = 325 nM T16633 D03VHX 44388111 IC50 = 25 nM T16633 D04EWA 44388034 IC50 = 535 nM T16633 D04FPW 44388024 IC50 = 720 nM T16633 D04ORV 44388047 IC50 = 5.3 nM T16633 D04QBM 5311374 IC50 > 1000 nM T16633 D05COQ 11847588 IC50 > 1000 nM T16633 D05XZA 44388071 IC50 = 14 nM T16633 D06JWT 44388073 IC50 = 75 nM T16633 D07DUF 44388130 IC50 = 248 nM T16633 D07OSF 44388044 IC50 = 583 nM T16633 D07WRP 15965425 Ki = 2392 nM T16633 D09DAC 44388046 IC50 = 59 nM T16633 D09LHN 44311674 IC50 = 15 nM T16633 D0A0DO 44388056 IC50 = 260 nM T16633 D0A1XX 44388113 IC50 = 45 nM T16633 D0BE3D 44388092 IC50 = 8 nM T16633 D0C5RH 44388125 IC50 = 112 nM T16633 D0CC1P 44388042 IC50 = 69 nM T16633 D0H0DC 44388051 IC50 > 1000 nM T16633 D0H4WH 44388128 IC50 = 0.98 nM T16633 D0I9ME 44388074 IC50 = 7.2 nM T16633 D0J5OY 44388022 IC50 = 79 nM T16633 D0M5LA 44388050 IC50 > 1000 nM T16633 D0N2MA 44388103 IC50 = 15 nM T16633 D0N4LH 44388065 IC50 = 151 nM T16633 D0O4GU 44403230 Ki > 1000 nM T16633 D0P6ZZ 10581102 IC50 > 1000 nM T16633 D0R0OX 44388102 IC50 = 16 nM T16633 D0R4IS 44388131 IC50 = 113 nM T16633 D0S7YR 44388059 IC50 = 14 nM T16633 D0T5RO 16129706 IC50 = 0.14 nM T16633 D0W0AF 44388072 IC50 = 10 nM T16633 D0WG0O 44388049 IC50 > 1000 nM T16633 D0Z0OF 44388094 IC50 = 2.5 nM T16633 D0Z1XY 44388064 IC50 = 23 nM T16633 D0Z3LZ 44388023 IC50 = 197 nM T65783 C2J1RE 351037 IC50 > 79000 nM T65783 CX9FV4 7217852 IC50 > 79000 nM T65783 CR1QE5 7217853 IC50 > 79000 nM T65783 C12BHY 7217856 IC50 > 79000 nM T65783 C86MDE 7217859 IC50 > 79000 nM T65783 C9UBG6 7217861 IC50 > 79000 nM T65783 C3XLA7 7217862 IC50 > 79000 nM T65783 C4Y6JF 7217867 IC50 > 79000 nM T65783 CB8NT2 7217870 IC50 > 79000 nM T65783 CT6F3C 7217876 IC50 > 79000 nM T65783 C8PK9D 7217878 IC50 > 79000 nM T65783 CYX8F6 7217879 IC50 > 79000 nM T65783 CH3I6U 7217884 IC50 > 79000 nM T65783 CI92NG 7217887 IC50 > 79000 nM T65783 C17GSL 7217891 IC50 > 79000 nM T65783 C1W3XE 7217912 IC50 > 79000 nM T65783 C8RWT6 7217913 IC50 > 79000 nM T65783 CFOJ16 7217916 IC50 > 59000 nM T65783 C5LZ0X 7217919 IC50 > 79000 nM T65783 CNG45O 7217921 IC50 = 54500 nM T65783 C2PQ8W 7217922 IC50 > 79000 nM T65783 CA7EW6 7217938 IC50 = 75700 nM T65783 CK9X8S 7217939 IC50 = 59200 nM T65783 CT89GV 7217942 IC50 = 3110 nM T65783 C07ZXA 7217944 IC50 = 72200 nM T65783 CUA9S4 7217946 IC50 = 7250 nM T65783 C7AMT6 7217947 IC50 = 4700 nM T65783 CCE5T6 7217950 IC50 = 29000 nM T65783 CW2AT7 7218011 IC50 > 79000 nM T65783 C9ZEC8 12005825 IC50 = 39900 nM T65783 C1D7HW 12005898 IC50 = 74100 nM T65783 C4K8HT 12005992 IC50 = 1750 nM T65783 CB78RO 16130452 EC50 = 1.9 nM T65783 C0A9WY 16194671 IC50 > 79000 nM T65783 C6J4NC 16805942 IC50 = 18200 nM T65783 C21UXH 16832372 IC50 > 79000 nM T65783 C9IP8D 18572334 IC50 > 79000 nM T65783 CK2L9R 18572335 IC50 = 58800 nM T65783 CO48HV 18572337 IC50 = 51000 nM T65783 CC70BA 18572338 IC50 = 6200 nM T65783 CMG17E 18572343 IC50 = 20600 nM T65783 CQ3ZV0 18572352 IC50 > 79000 nM T65783 CZ2FW0 18572378 IC50 > 79000 nM T65783 COP52X 18572379 IC50 > 79000 nM T65783 CAJH61 18572382 IC50 > 79000 nM T65783 CNKA87 18572395 IC50 > 79000 nM T65783 C27ZCA 25085173 EC50 = 0.0122 nM T65783 C8TX1U 42281625 IC50 > 79000 nM T65783 CB31ST 44726831 IC50 > 79000 nM T65783 CH41CI 46835118 IC50 > 79000 nM T65783 C5LJ0V 46835120 IC50 > 79000 nM T65783 CSBO37 46835124 IC50 > 79000 nM T65783 C6EFX7 46905014 IC50 > 79000 nM T65783 CCUA93 46905018 IC50 = 8510 nM T65783 C85DJM 46905020 IC50 > 79000 nM T65783 CBNT43 46905022 IC50 > 79000 nM T65783 CH20YA 46905025 IC50 > 79000 nM T65783 CWER26 46905028 IC50 = 9610 nM T65783 CD3CK1 46905029 IC50 = 6590 nM T65783 CU6D2Q 46905034 IC50 = 3210 nM T65783 CWY35N 46905037 IC50 > 79000 nM T65783 CP3M2F 46905038 IC50 > 79000 nM T65783 CQK7D4 49787115 IC50 > 79000 nM T65783 C86OIB 49787117 IC50 > 79000 nM T65783 CL3D2B 49787119 IC50 > 79000 nM T65783 CP5M7Y 49787120 IC50 > 79000 nM T65783 CW9G1R 49842899 IC50 = 24000 nM T65783 CVC2N3 49842902 IC50 = 4530 nM T65783 C9T3AM 49842903 IC50 = 8270 nM T65783 CQ6V4E 49842905 IC50 = 12800 nM T65783 C62CDL 49842908 IC50 > 79000 nM T65783 CCQK74 71456693 IC50 > 79000 nM T65783 CGM32X 71462076 IC50 > 79000 nM T65783 C0DO6L 90644396 EC50 > 30000 nM T65783 CWY43T 90644398 EC50 > 30000 nM T65783 CM1HI5 90656606 EC50 = 237 nM T65783 CEA07I 90656607 EC50 = 494 nM T65783 CKF15X 90656608 EC50 = 539 nM T65783 C6V8TM 90656609 EC50 = 637 nM T65783 CO51PF 90656610 EC50 = 691 nM T65783 C7QO0V 90656611 EC50 = 936 nM T65783 C2Q6JA 90656612 EC50 = 1383 nM T65783 C34OGA 90656613 EC50 = 2350 nM T65783 C7V8EM 90656614 EC50 > 3000 nM T65783 CXRO89 90656615 EC50 > 3000 nM T65783 CBAT91 90656616 EC50 > 3000 nM T65783 C8SH3Y 90656617 EC50 > 3000 nM T65783 C18FEA 90656618 EC50 > 3000 nM T65783 CSO54R 90656619 EC50 > 3000 nM T65783 CQ41HU 90656620 EC50 = 1.1 nM T65783 CU9WH0 90656621 EC50 = 1.7 nM T65783 CUP8F7 90656622 EC50 = 1.9 nM T65783 CDIT19 90656623 EC50 = 2.2 nM T65783 C8X2RV 90656624 EC50 = 3.2 nM T65783 C3ZYS4 90656625 EC50 = 4.4 nM T65783 C40WHE 90656626 EC50 = 4.7 nM T65783 CB3FP8 90656627 EC50 = 8.9 nM T65783 CS24BV 90656628 EC50 = 19 nM T65783 CB3GE1 90656629 EC50 = 20 nM T65783 CPM9T5 90656630 EC50 = 31 nM T65783 CF2K0U 90656631 EC50 = 33 nM T65783 C42XWN 90656632 EC50 = 44 nM T65783 CIG7P5 90656633 EC50 = 73 nM T65783 C4J2ZT 90656634 EC50 > 31622.78 nM T65783 C6A0XD 90656635 EC50 > 31622.78 nM T65783 C7CAH3 90656636 EC50 = 83.18 nM T65783 CH95OZ 118568543 EC50 > 30000 nM T65783 CW49MU 118568545 EC50 > 30000 nM T65783 CDN05V 118568560 EC50 > 30000 nM T65783 C1C2IW 118568561 EC50 > 30000 nM T65783 C9FZ8G 118568562 EC50 > 30000 nM T65783 C28JSA 118568565 EC50 > 30000 nM T65783 CMT3D1 118568636 EC50 > 30000 nM T65783 CI69JT 118568646 Ki = 600 nM T65783 C3XF1J 118568676 EC50 > 30000 nM T65783 C12TDY 118568780 EC50 > 30000 nM T65783 CL0J9I 118568782 EC50 > 30000 nM T65783 CJ5PN1 118568784 EC50 > 30000 nM T65783 C63ZXV 118568855 EC50 > 30000 nM T65783 C52VYU 118568856 EC50 > 30000 nM T65783 CR2Z9X 118568860 EC50 > 30000 nM T65783 C2M3GZ 118568863 EC50 > 30000 nM T65783 CUL40R 118568915 EC50 > 30000 nM T65783 C04CFZ 118568917 EC50 > 30000 nM T65783 CAGX81 118568919 EC50 > 30000 nM T65783 CMZ87V 118568922 EC50 > 30000 nM T65783 CS9PK1 118568930 EC50 > 30000 nM T65783 CUV5Y0 118715454 EC50 = 33.7 nM T65783 C6GV2L 118715455 EC50 > 30000 nM T65783 CQ1DR4 118715456 EC50 > 30000 nM T65783 C7BI9F 118715457 EC50 = 198.6 nM T65783 C7LC0E 118715458 EC50 = 41.3 nM T65783 CZHB45 118715459 EC50 > 30000 nM T65783 C3W1VQ 118715460 EC50 > 30000 nM T65783 CD89JW 118715461 EC50 > 30000 nM T65783 CAJ0T1 118715462 EC50 > 30000 nM T65783 C6VR9K 118715463 EC50 = 21.5 nM T65783 C9H6VU 118715464 EC50 = 95.7 nM T65783 CSJV63 118715465 EC50 > 30000 nM T65783 C80LTN 118715466 EC50 = 2.7 nM T65783 CJB6N8 118715467 EC50 > 30000 nM T65783 CS2V3H 118715468 EC50 > 30000 nM T65783 CML9P4 118715469 EC50 > 30000 nM T65783 C5WPH4 118715470 EC50 > 30000 nM T65783 C9OE3S 118715471 EC50 > 30000 nM T65783 CWX0L5 118715472 EC50 > 30000 nM T65783 C5N6XM 118715473 EC50 > 30000 nM T65783 CAJS62 118715474 EC50 > 30000 nM T65783 C9GU6K 118715475 EC50 > 30000 nM T65783 C0GEY6 118715476 EC50 > 30000 nM T65783 CXN6C1 118715477 EC50 = 225.5 nM T65783 CM5L8N 118715478 EC50 > 30000 nM T65783 CK4BT2 118715479 EC50 > 30000 nM T65783 CGRB51 118734703 EC50 = 0.53 nM T65783 C1LI8R 118734704 EC50 = 2.5 nM T65783 C8C5KO 118734767 EC50 = 1.3 nM T65783 C9ZWT7 118734768 EC50 = 2.7 nM T65783 C2H6BG 118734769 EC50 = 0.23 nM T65783 C63JPQ 118734770 EC50 = 0.17 nM T65783 C8H7JV 118734771 EC50 = 0.45 nM T65783 CSB8T7 118734772 Ki = 1.3 nM T65783 CT4AL0 118734773 EC50 = 3 nM T65783 C16IYO 118734774 EC50 = 2.7 nM T65783 CWG68D 118734775 EC50 = 0.24 nM T65783 CI8X3T 118734776 Ki = 0.016 nM T65783 C0S4AY 118734777 EC50 = 0.04 nM T65783 C87ZQV 118734778 EC50 = 0.63 nM T65783 C43YQF 118734779 EC50 = 6 nM T65783 CD8K0G 118734780 EC50 = 1.3 nM T65783 CBP0F2 118734781 EC50 = 0.07 nM T65783 C6FE7W 118734782 Ki = 0.69 nM T65783 CDS7I4 118734783 EC50 = 1.1 nM T65783 C4D3ZK 118734784 Ki = 46 nM T65783 CVD6R8 118734785 Ki > 10000 nM T65783 C3SVZ9 118734786 Ki > 10000 nM T65783 CZ93DF 118734787 Ki > 10000 nM T65783 CY4IS2 127043374 EC50 = 0.1175 nM T65783 CG0B6M 127044072 Ki = 11 nM T65783 CV98XE 127044698 Ki = 0.53 nM T65783 C0AQ2M 127045179 EC50 = 36 nM T65783 C1DOZ7 127045180 Ki = 3.4 nM T65783 C7PG9N 127045189 Ki = 8.4 nM T65783 CAYI14 127048431 EC50 > 30000 nM T65783 C3WSB4 127051011 Ki = 1400 nM T65783 CI1WH7 127051222 Ki = 3000 nM T65783 CNUA86 127051280 EC50 = 800 nM T65783 CR9PV6 127052214 EC50 > 30000 nM T65783 C45ZLA 134828250 EC50 = 0.2884 nM T65783 CM3L9F 137224964 EC50 > 30000 nM T65783 CB3N6E 137225067 EC50 > 30000 nM T65783 CD1OV6 137501999 EC50 = 0.093 nM T65783 C54VFS 137502080 EC50 = 0.083 nM T65783 CU62XA 137502125 EC50 = 1.4 nM T65783 CN5KB9 137502168 EC50 = 7.4 nM T65783 CKW9L0 137631382 Ki = 188 nM T65783 C3Z0OT 137632615 EC50 = 4.9 nM T65783 C48ZSL 137633995 Ki = 523 nM T65783 CB1WI7 137635080 Ki = 194 nM T65783 CI0BM8 137638986 Ki = 6074 nM T65783 C3TN2R 137639006 EC50 = 0.8 nM T65783 C0BFG1 137639727 Ki = 1.9 nM T65783 CG3IH1 137641320 Ki = 917 nM T65783 CJN34B 137643637 Ki = 14 nM T65783 CGXF65 137645721 Ki = 41 nM T65783 C6M1DB 137646730 Ki = 3 nM T65783 CIR0E2 137647010 Ki = 2.9 nM T65783 CNM5T3 137649041 Ki = 0.1 nM T65783 CB9TJ2 137649272 Ki = 5.7 nM T65783 CDC79S 137649320 EC50 = 0.4 nM T65783 CYN21T 137649702 Ki = 509 nM T65783 CYJ61K 137649936 Ki = 206 nM T65783 C1R2JM 137650169 EC50 = 2.1 nM T65783 C8UPE0 137650201 Ki = 310 nM T65783 C7E3TJ 137650464 Ki = 0.3 nM T65783 C2FNP8 137650548 Ki = 1.4 nM T65783 C78RKA 137650891 Ki = 445 nM T65783 C3OI7C 137650935 Ki = 1.1 nM T65783 C6PJB4 137651612 Ki = 489 nM T65783 C2EYV9 137652055 Ki > 10000 nM T65783 C9XIL8 137653279 Ki = 41 nM T65783 C64CAP 137654306 Ki = 268 nM T65783 C12MDR 137654459 EC50 = 2 nM T65783 C8E4TP 137654488 Ki = 0.15 nM T65783 CHS13O 137657220 Ki = 3.9 nM T65783 CZ2W4O 137657369 Ki > 10000 nM T65783 CH1TJ2 137658661 Ki = 9.1 nM T65783 CP93BF 137660518 Ki = 4.5 nM T65783 CZF97Q 137661816 EC50 = 4.1 nM T65783 C59HBK 145948593 Ki = 0.14 nM T65783 CZ2AO7 145948594 EC50 = 22 nM T65783 CA0RT3 145948599 Ki = 0.37 nM T65783 CZF6H8 145948600 Ki = 14 nM T65783 CJ2RY1 145948634 Ki = 0.93 nM T65783 CU2QW4 145948635 Ki = 0.19 nM T65783 C71CST 145948636 Ki = 0.14 nM T65783 C1QLU9 145948641 Ki = 6.8 nM T65783 C35JCH 145948642 Ki = 0.84 nM T65783 CE97TL 145948643 EC50 = 147 nM T65783 C8RW6H 145948663 Ki = 4 nM T65783 C8W0LA 145948664 EC50 = 19 nM T65783 CXY19O 145948665 Ki = 0.23 nM T65783 C27DKH 145948668 Ki = 48 nM T65783 C3CYU6 145948669 EC50 = 20 nM T65783 CG74BR 145948671 Ki = 0.34 nM T65783 CHZI56 145948672 Ki = 20 nM T65783 C81UGK 154603299 EC50 = 0.18 nM T65783 CXI28P 154603335 EC50 = 0.31 nM T65783 COES94 154603343 EC50 = 19 nM T65783 CYT83N 154603359 EC50 = 0.51 nM T65783 CKY36L 154603363 EC50 = 1.5 nM T65783 CE3Q6L 154603384 EC50 = 9 nM T65783 CCD21A 154603387 EC50 = 5.7 nM T65783 C9O1UP 154603393 EC50 = 5.7 nM T65783 CE17OJ 154603397 EC50 = 0.6 nM T65783 CLY4A3 154995949 EC50 = 0.062 nM T65783 CQ8LU1 155004167 EC50 = 51 nM T65783 CX7G0Z 155513131 EC50 = 50 nM T65783 C8D1MN 155514255 EC50 = 176 nM T65783 CNS13I 155514812 EC50 = 11.3 nM T65783 C2F4BN 155515730 EC50 = 29 nM T65783 C6PD7V 155516838 EC50 = 2.7 nM T65783 CSH8L0 155516953 EC50 = 0.19 nM T65783 CEF4W2 155529276 EC50 = 0.1 nM T65783 C1NCA3 155530998 EC50 = 6.3 nM T65783 CSO3T4 155536031 EC50 = 2.5 nM T65783 C5WY4V 155543212 EC50 = 4900 nM T65783 CO0PQ5 155550782 EC50 = 2.6 nM T65783 CRV3E4 155553677 EC50 = 59 nM T65783 CJ68GT 155557915 EC50 = 568 nM T65783 C8AWJ3 155558340 EC50 = 2100 nM T65783 C1PQR8 155566712 EC50 = 0.33 nM T65783 D00QYH 25078060 EC50 = 0.87 nM T65783 D05NXX 7217941 IC50 = 700 nM T65783 D0I8TR 46905036 EC50 = 3700 nM T98933 D0L5WM 2157 IC50 = 600 nM T98933 D0S6JG 5920 Ki = 0.08 nM T98933 D0Z4EI 55245 Ki > 2250 nM T98933 D01QXY 9862248 Ki = 0.32 nM T98933 D03MYO 15981237 EC50 = 210 nM T98933 D07ZTD 15942005 Ki = 600 nM T98933 D0J6XC 5803 IC50 = 0.048 nM T98933 D0V5FQ 166559 Ki = 2.17 nM T98933 D02WGY 10299876 Ki = 0.43 nM T98933 D07EGS 9874938 Ki = 0.47 nM T98933 CNJ29A 861 IC50 = 0.103 nM T98933 CLSK17 5804 IC50 = 0.019 nM T98933 C47GSU 79170 IC50 = 9100 nM T98933 C40JPQ 447271 Ki = 0.03 nM T98933 C57HCR 652088 IC50 = 69800 nM T98933 CB6HQ4 656928 IC50 = 0.6166 nM T98933 CG59SJ 2404806 IC50 = 23100 nM T98933 CJN3P5 4266779 IC50 = 16500 nM T98933 CU1I3O 4652254 IC50 > 100000 nM T98933 C3S6ZI 5184800 IC50 = 4100 nM T98933 C79ZDX 5287525 IC50 = 175 nM T98933 C6ZXJ7 6431911 IC50 = 0.1096 nM T98933 CRQ1O4 9819350 Ki = 0.5 nM T98933 C4PCB9 9825337 EC50 = 49 nM T98933 CZ4I9T 9828296 Ki = 0.46 nM T98933 CQR6U0 9838979 IC50 = 47 nM T98933 C3MZ1Y 9843007 Ki = 7.8 nM T98933 CJ6E2M 9847869 Ki = 0.63 nM T98933 CA27CJ 9862799 IC50 = 20.89 nM T98933 CZ82PF 9863447 Ki = 0.24 nM T98933 CC64MT 9869395 IC50 = 910 nM T98933 CZ1U7X 9932398 IC50 = 2.089 nM T98933 CY01RH 9933119 IC50 = 0.095 nM T98933 CHG6L7 9933993 IC50 = 18 nM T98933 CFS8T0 9944477 IC50 = 2620 nM T98933 C46NXU 9951790 Ki = 0.06 nM T98933 CFH9D2 9968513 IC50 = 1300 nM T98933 CN30MV 9980009 EC50 = 500 nM T98933 CX4MZ9 9980722 IC50 = 1.8 nM T98933 CZ96GN 10030727 IC50 = 12 nM T98933 CJ05DK 10049652 IC50 = 1.8 nM T98933 CP1R7A 10113366 IC50 = 120 nM T98933 CY8S9M 10133886 IC50 = 110 nM T98933 C72HTV 10135986 IC50 = 520 nM T98933 CMY69T 10137392 IC50 = 360 nM T98933 CGE9I7 10151760 Ki = 8.2 nM T98933 CUC0Y8 10172901 Ki = 59 nM T98933 C1Y3FJ 10174187 Ki = 6 nM T98933 CD4SX7 10202877 IC50 = 820 nM T98933 CNPD04 10216950 Ki = 1.19 nM T98933 CDY6F5 10238439 Ki = 3.7 nM T98933 C1DYU9 10269704 Ki = 10 nM T98933 CJB2E3 10274474 Ki = 0.4 nM T98933 C7UYX0 10276774 Ki = 0.5 nM T98933 CH5NX1 10279835 Ki = 2 nM T98933 CW26FQ 10287060 Ki = 2.59 nM T98933 CIB52S 10297431 IC50 = 141.25 nM T98933 CSC3T4 10299993 IC50 = 15.85 nM T98933 C81BSZ 10309431 Ki = 15.1 nM T98933 C09IJX 10310671 Ki = 57.6 nM T98933 CT13FC 10310672 Ki = 53.5 nM T98933 C0VMH3 10321482 IC50 = 680 nM T98933 C7TGL0 10322653 Ki = 0.51 nM T98933 CN3G5V 10390904 Ki = 0.07 nM T98933 CL81KF 10413582 EC50 = 380 nM T98933 CP8O0Q 10455127 IC50 = 13 nM T98933 C3UAD9 10456672 IC50 = 0.3 nM T98933 C5N7BD 10456830 IC50 = 0.025 nM T98933 C34MFS 10457976 IC50 = 22 nM T98933 C4T6ZH 10479778 IC50 = 0.3 nM T98933 CM4ED8 10479779 IC50 = 0.28 nM T98933 CU42IL 10897325 IC50 = 4000 nM T98933 CX2RY1 10904700 IC50 = 0.1514 nM T98933 CZ3SX1 10918755 IC50 = 480 nM T98933 CD9G7N 11164881 IC50 = 1819.7 nM T98933 C6OX1A 11209929 IC50 = 32000 nM T98933 CPY31C 11247142 IC50 = 120 nM T98933 CA8Z1T 11281247 IC50 = 810 nM T98933 CY0M1L 11395277 IC50 = 1800 nM T98933 C48UZO 11463526 IC50 = 700 nM T98933 C5CZ2Q 11998611 Ki = 14600 nM T98933 CRJ1N9 11999781 Ki = 2.5 nM T98933 C7N4HR 11999783 Ki = 1.51 nM T98933 CW01OG 12001110 EC50 = 40 nM T98933 C1AU0V 13958302 Ki = 238 nM T98933 CDB93J 15219550 IC50 = 17700 nM T98933 CDKZ56 15940421 Ki = 42.1 nM T98933 CM17XO 15941848 Ki = 2.17 nM T98933 C1QZ3U 15941849 Ki = 36 nM T98933 CRK5V2 15941850 Ki = 271 nM T98933 C7PV1O 15941997 Ki = 2.51 nM T98933 C7BD0S 15941998 Ki = 30.5 nM T98933 C93MUZ 15942131 Ki = 6.64 nM T98933 CNCW45 15942413 Ki = 9.1 nM T98933 CEQ1J5 15981204 EC50 = 7750 nM T98933 CZEJ29 15981205 EC50 = 7010 nM T98933 C47AYJ 15981206 EC50 = 460 nM T98933 CRF9T7 15981207 EC50 = 2380 nM T98933 C4XF0E 15981234 EC50 = 700 nM T98933 C7U4OQ 15981235 EC50 = 670 nM T98933 CT9N6B 15981236 EC50 = 120 nM T98933 CTI37Q 15981238 EC50 = 120 nM T98933 CIM62O 15981239 EC50 = 770 nM T98933 CB6UE5 15981240 EC50 = 220 nM T98933 CL0FG1 15981241 EC50 = 90 nM T98933 C4BU2G 15981272 EC50 = 2990 nM T98933 C5BO7H 15981273 EC50 = 600 nM T98933 CES0V2 15981274 EC50 = 2040 nM T98933 CCKG05 15981275 EC50 = 9170 nM T98933 C2SR1B 15981276 EC50 = 6980 nM T98933 CIB52A 15981279 EC50 = 140 nM T98933 CWK35C 16730429 IC50 = 60 nM T98933 C7G2AM 18415120 Ki = 15.5 nM T98933 CD0L4R 21110667 Ki = 12 nM T98933 C0AQU8 21110669 Ki = 30 nM T98933 CZI6V2 21110670 Ki = 41 nM T98933 C47HQO 21110672 Ki = 40 nM T98933 CV3FE0 21110673 Ki = 17 nM T98933 CCGP69 21110677 Ki = 53.6 nM T98933 CM0DL5 21110680 Ki = 81.3 nM T98933 CHN91T 21110689 Ki = 39.9 nM T98933 CHT5Y9 21110691 Ki = 19.7 nM T98933 C7TN9A 21110692 Ki = 40.2 nM T98933 CX5I2A 21636517 IC50 = 66000 nM T98933 C6TCO8 21992496 IC50 = 1320 nM T98933 C5EFH7 21992497 IC50 = 88 nM T98933 CO3X7S 21992575 IC50 = 48 nM T98933 COV0S9 21992584 IC50 = 121 nM T98933 CVD9T3 21992651 IC50 = 646 nM T98933 C0QS8C 21992678 IC50 = 78 nM T98933 C5N7DG 21992681 IC50 = 343 nM T98933 CSY41F 21992749 IC50 = 4000 nM T98933 CTF0Q7 21992824 IC50 = 877 nM T98933 C7KTU1 21992839 IC50 = 9290 nM T98933 C6QNL9 21992913 IC50 = 71 nM T98933 CNF16U 22339386 Ki = 0.1 nM T98933 CF2X6V 22339458 Ki = 0.04 nM T98933 CD08GC 22339531 Ki = 0.72 nM T98933 C3HMF6 22339537 Ki = 13 nM T98933 CF7ZI8 22339599 Ki = 0.64 nM T98933 CASB98 22339607 Ki = 1.9 nM T98933 CNLT41 22339633 Ki = 0.13 nM T98933 C89IYX 22339645 Ki = 0.02 nM T98933 CV57KF 22339648 Ki = 27 nM T98933 CY2HZ3 22339678 IC50 = 0.6457 nM T98933 CWV5B9 22339727 Ki = 0.4 nM T98933 CK0C8N 22339743 Ki = 0.46 nM T98933 CF2CQ7 22372339 IC50 = 61000 nM T98933 CR7DC6 23546124 IC50 = 104 nM T98933 CFV3P7 23635238 IC50 = 1500 nM T98933 CWE74Y 23635239 IC50 = 1600 nM T98933 CM6S4G 23635240 IC50 = 2000 nM T98933 CPR67K 23635363 IC50 = 3900 nM T98933 CI6D4Y 23635365 IC50 = 12100 nM T98933 CAHT12 23635366 IC50 = 12700 nM T98933 C1G2TO 23635477 IC50 = 23200 nM T98933 C17PKJ 23635478 IC50 > 100000 nM T98933 CC3VU5 23635479 IC50 > 100000 nM T98933 CGU3Z0 23635480 IC50 > 100000 nM T98933 C82WJG 23635600 IC50 = 55800 nM T98933 C18SZO 23635729 IC50 = 20300 nM T98933 C7BLC2 23635731 IC50 > 100000 nM T98933 CE6DP7 23635732 IC50 > 100000 nM T98933 CGL6T0 23635852 IC50 > 100000 nM T98933 CK4XI2 23635853 IC50 > 100000 nM T98933 CY80FR 23635854 IC50 > 100000 nM T98933 C7NAV1 23635855 IC50 = 35100 nM T98933 CU81CL 23635857 IC50 > 100000 nM T98933 C31FPX 23635859 IC50 > 100000 nM T98933 CQ2E7G 23642624 IC50 = 85900 nM T98933 CB38IZ 23644731 IC50 = 67.61 nM T98933 CT5QC3 23648079 IC50 = 0.11 nM T98933 CP7SV3 23648080 IC50 = 2.7 nM T98933 CYU20W 23648081 IC50 = 1.3 nM T98933 C3V1BH 23648082 IC50 = 5.9 nM T98933 C1JIZ5 23648083 IC50 = 0.27 nM T98933 C3QR1F 23648084 IC50 = 0.71 nM T98933 C0N2YD 23648085 IC50 = 0.78 nM T98933 C08JWQ 23648086 IC50 = 0.6 nM T98933 C5INJ3 23648087 IC50 = 290 nM T98933 CTJK20 23648089 IC50 = 1400 nM T98933 CE4R6V 23648090 IC50 = 2600 nM T98933 C84TAV 23648093 IC50 = 200 nM T98933 CB7OK8 23648094 IC50 = 160 nM T98933 C45JQX 23648095 IC50 = 190 nM T98933 C80CEB 23648096 IC50 = 87 nM T98933 CV20UI 23648101 IC50 = 0.1995 nM T98933 CIKD57 23648102 IC50 = 4.266 nM T98933 CV91YT 23648103 IC50 = 46.77 nM T98933 C5WKV2 23648104 IC50 = 44.67 nM T98933 C5V6OQ 23648105 IC50 = 2.884 nM T98933 C91FSP 23648106 IC50 = 3.236 nM T98933 CBD9J5 23648107 IC50 = 0.8511 nM T98933 C3R0GX 23648108 IC50 = 67.61 nM T98933 C1SXM0 23648109 IC50 = 3.981 nM T98933 C98FIL 23648110 IC50 = 20.89 nM T98933 C7R2XE 23648111 IC50 = 10.96 nM T98933 CR85SZ 23648112 IC50 = 0.7762 nM T98933 CN2YX0 23648113 IC50 = 3.388 nM T98933 CC69AB 23648114 IC50 = 50.12 nM T98933 COP12V 23648115 IC50 = 75.86 nM T98933 CN5T8D 23648116 IC50 = 87.1 nM T98933 C7ON2Q 23648118 IC50 = 40.74 nM T98933 CTR20F 23648121 IC50 = 7.762 nM T98933 CXTZ50 23648122 IC50 = 6.026 nM T98933 CZ8J0T 23648123 IC50 = 7.586 nM T98933 C12HDM 23648124 IC50 = 1.096 nM T98933 C0UJ6X 23648125 IC50 = 9.55 nM T98933 CFA1Y6 23648126 IC50 = 60.26 nM T98933 C35AZQ 23648127 IC50 = 83.18 nM T98933 CR1S4E 23648128 IC50 = 46.77 nM T98933 C0WY3I 23648129 IC50 = 6.026 nM T98933 CL60SF 23648130 IC50 = 34.67 nM T98933 C72TJZ 23648131 IC50 = 4.169 nM T98933 COL8Q7 23648132 IC50 = 6.761 nM T98933 CNWC43 23648133 IC50 = 18.2 nM T98933 C4SW8I 23648134 IC50 = 4.786 nM T98933 CQ7M3I 23648135 IC50 = 4.898 nM T98933 CQW43F 23648136 IC50 = 8.511 nM T98933 C62YFJ 23648137 IC50 = 37.15 nM T98933 CICP87 23648138 IC50 = 67.61 nM T98933 CWT25S 23648139 IC50 = 3.467 nM T98933 C5XD8Q 24830528 IC50 = 40 nM T98933 CR2A9H 24830680 EC50 = 220 nM T98933 CD6EI3 24830686 EC50 = 190 nM T98933 CKDP62 24830833 EC50 = 1300 nM T98933 CO9E2H 24894049 EC50 = 317 nM T98933 C5BS8M 25149230 Ki = 26 nM T98933 CJ6LC2 25149503 Ki = 9.72 nM T98933 CT0J6H 25149504 Ki = 106 nM T98933 CFW74J 25149505 Ki = 146 nM T98933 C5MFE8 25149592 Ki = 52.3 nM T98933 CLSD47 25149598 Ki = 25.4 nM T98933 CZP70F 25150124 Ki = 89.7 nM T98933 C4MT7I 25150127 Ki = 87 nM T98933 C7G5CL 25150225 Ki = 128 nM T98933 C57AUE 25150325 Ki = 0.84 nM T98933 CLZ86A 25150424 Ki = 0.97 nM T98933 CRW82I 44136896 IC50 = 430 nM T98933 C2Y6AG 44185845 IC50 = 1100 nM T98933 COT19A 44185854 IC50 = 600 nM T98933 CSQ1C0 44185855 IC50 = 1700 nM T98933 CTG0X6 44185856 IC50 = 1100 nM T98933 C1L8KQ 44185857 IC50 = 1100 nM T98933 C2VWY6 44185858 IC50 = 5300 nM T98933 CXF3N9 44185859 IC50 = 11200 nM T98933 C8GIP0 44185860 IC50 = 4000 nM T98933 CC4E7U 44185914 IC50 = 4200 nM T98933 CMS09A 44185915 IC50 = 600 nM T98933 C1GI8D 44185916 IC50 = 500 nM T98933 CQAT73 44186032 IC50 = 7100 nM T98933 CC0YN9 44186033 IC50 > 50000 nM T98933 C7VZI4 44186034 IC50 = 10100 nM T98933 CR1D9P 44186035 IC50 = 5300 nM T98933 CC32IS 44186097 IC50 = 7000 nM T98933 C2MG6T 44186098 IC50 = 25300 nM T98933 C4XV1B 44186099 IC50 = 5100 nM T98933 CFJ0P8 44186100 IC50 > 50000 nM T98933 C31NSX 44186101 IC50 = 4700 nM T98933 CBM5Z6 44186102 IC50 = 1800 nM T98933 CX10SK 44186103 IC50 = 2600 nM T98933 C8TU3K 44186104 IC50 = 2700 nM T98933 CWY0A2 44186168 IC50 = 8400 nM T98933 CO65HR 44186169 IC50 = 2700 nM T98933 C1TU5I 44186170 IC50 = 1900 nM T98933 CC49MP 44186171 IC50 = 5000 nM T98933 C3M4KR 44186172 IC50 = 1790 nM T98933 C4COU6 44186173 IC50 = 600 nM T98933 CPZ6T3 44186174 IC50 = 690 nM T98933 C40ENX 44186175 IC50 > 50000 nM T98933 CIL71S 44186232 IC50 > 50000 nM T98933 CP1A5G 44186233 IC50 > 50000 nM T98933 C4CMU9 44186234 IC50 > 50000 nM T98933 CM9V8Z 44186235 IC50 = 1700 nM T98933 CDI86U 44186236 IC50 = 1600 nM T98933 C2YL8N 44186237 IC50 = 18900 nM T98933 CYO36K 44186238 IC50 = 22000 nM T98933 CRHL62 44186239 IC50 = 3800 nM T98933 CS2N6F 44186298 IC50 > 50000 nM T98933 CES48R 44186299 IC50 > 50000 nM T98933 C6XEM3 44186300 IC50 > 50000 nM T98933 C35QER 44186301 IC50 > 50000 nM T98933 CREP27 44186302 IC50 > 50000 nM T98933 CPLW35 44186303 IC50 = 4900 nM T98933 C1PFT0 44186305 IC50 > 50000 nM T98933 C5A1HF 44186364 IC50 = 4600 nM T98933 C6PW0U 44186365 IC50 = 4800 nM T98933 CYE39G 44186366 IC50 = 1200 nM T98933 CS6MG3 44186367 IC50 = 5000 nM T98933 C7CP9D 44186368 IC50 = 1200 nM T98933 CC35ST 44186369 IC50 = 1200 nM T98933 CA62XQ 44186370 IC50 = 5000 nM T98933 C1O4YR 44186418 IC50 = 2000 nM T98933 CYH8U5 44186419 IC50 = 1700 nM T98933 C95GQS 44186420 IC50 = 800 nM T98933 CA1EV7 44186421 IC50 = 10400 nM T98933 CU64OD 44186422 IC50 = 5000 nM T98933 C9J0YD 44186423 IC50 = 4300 nM T98933 C25UOE 44186424 IC50 = 1400 nM T98933 CX9U3Q 44186425 IC50 = 2100 nM T98933 CTF94W 44186465 IC50 = 1500 nM T98933 C9G8JS 44186466 IC50 = 800 nM T98933 C7TFN6 44186467 IC50 = 2000 nM T98933 CD2UC4 44186468 IC50 = 1900 nM T98933 C0Z9OK 44186469 IC50 = 2400 nM T98933 CTJ1O5 44186470 IC50 = 3000 nM T98933 CN8QS2 44186471 IC50 = 700 nM T98933 C78TSP 44186472 IC50 = 1100 nM T98933 CL17KI 44186473 IC50 = 14100 nM T98933 COL0S6 44186474 IC50 = 4000 nM T98933 C75UOJ 44186475 IC50 > 50000 nM T98933 C1KVH2 44186476 IC50 > 50000 nM T98933 CK58UR 44186510 IC50 = 5400 nM T98933 CF1CU6 44186511 IC50 = 2000 nM T98933 CQB3X5 44186512 IC50 = 1700 nM T98933 C01ARC 44186513 IC50 = 1300 nM T98933 C7T3SZ 44186514 IC50 = 1300 nM T98933 CI27LX 44186515 IC50 = 900 nM T98933 C3DOF6 44186516 IC50 = 1200 nM T98933 C3SH2I 44186517 IC50 = 2300 nM T98933 C8X1EA 44186518 IC50 = 2700 nM T98933 CS7K3Y 44186519 IC50 = 5600 nM T98933 CHW5K6 44186520 IC50 > 50000 nM T98933 C58YWK 44186521 IC50 > 50000 nM T98933 CJPO14 44186523 IC50 = 5900 nM T98933 C3JN6A 44186555 IC50 = 4000 nM T98933 CUN70K 44186556 IC50 = 1000 nM T98933 C7CQN6 44186557 IC50 = 800 nM T98933 C9RI1Q 44186558 IC50 = 700 nM T98933 CP26OY 44186559 IC50 = 2400 nM T98933 C7FRJ9 44186560 IC50 = 1700 nM T98933 CB6C9M 44186561 IC50 = 1300 nM T98933 C2NPV9 44186562 IC50 = 12400 nM T98933 CYH38F 44186563 IC50 > 50000 nM T98933 C9G8SO 44186564 IC50 = 1800 nM T98933 C05IDW 44186565 IC50 = 2000 nM T98933 C73VSR 44186566 IC50 = 700 nM T98933 C3PH5N 44186567 IC50 = 600 nM T98933 C1F2WL 44186568 IC50 = 1400 nM T98933 CS6UN0 44186600 IC50 = 1600 nM T98933 CX5B3F 44186601 IC50 = 900 nM T98933 C9BJU8 44186602 IC50 = 3600 nM T98933 CE5MK1 44186603 IC50 = 2300 nM T98933 C1INA4 44186604 IC50 = 700 nM T98933 C60ECM 44186605 IC50 = 400 nM T98933 CM83FC 44186606 IC50 = 2900 nM T98933 CG2R8S 44186607 IC50 = 800 nM T98933 CM1UB2 44186608 IC50 = 4700 nM T98933 CWM3R1 44186609 IC50 = 600 nM T98933 CG2CH3 44186610 IC50 = 6500 nM T98933 CZQ2R1 44186611 IC50 = 18900 nM T98933 CFL30A 44186612 IC50 = 1500 nM T98933 C47SCQ 44186613 IC50 = 800 nM T98933 CZ7NW3 44186644 IC50 = 1500 nM T98933 CL52WN 44186645 IC50 = 700 nM T98933 CA5G8T 44186646 IC50 = 800 nM T98933 CEFM37 44186647 IC50 = 900 nM T98933 CK7N3X 44186648 IC50 = 1700 nM T98933 CE3JB8 44186649 IC50 = 600 nM T98933 CU7SG1 44186650 IC50 = 800 nM T98933 CI15SG 44186651 IC50 = 600 nM T98933 CY7VW4 44186652 IC50 = 3600 nM T98933 C0Q9AK 44186653 IC50 = 800 nM T98933 C0UL7Z 44186654 IC50 = 1200 nM T98933 C2ZF4S 44186655 IC50 = 1000 nM T98933 CKX1Q9 44186656 IC50 = 2100 nM T98933 C29QCE 44186657 IC50 = 900 nM T98933 CZQ7K2 44186691 IC50 = 800 nM T98933 CM80OW 44186692 IC50 = 700 nM T98933 C7OMH6 44186693 IC50 = 800 nM T98933 CQN2T6 44186694 IC50 = 3500 nM T98933 C0F2ZJ 44186695 IC50 = 5400 nM T98933 C63VSR 44186696 IC50 = 1500 nM T98933 C25FXN 44186698 IC50 = 800 nM T98933 CS0PI6 44186699 IC50 = 2100 nM T98933 C9PL4W 44186700 IC50 = 1000 nM T98933 C2ZEL5 44186701 IC50 = 1100 nM T98933 CO8R6C 44186702 IC50 = 900 nM T98933 CD0NW3 44186703 IC50 = 1200 nM T98933 C89HNC 44186704 IC50 = 700 nM T98933 C8UD7E 44299535 Ki = 2 nM T98933 CWH5G9 44345925 IC50 = 151 nM T98933 CQVW76 44346052 IC50 = 54 nM T98933 C87MEG 44346063 IC50 = 19500 nM T98933 C06YNJ 44349518 Ki = 0.16 nM T98933 CYAM86 44349526 Ki = 10000 nM T98933 CGXM40 44349576 Ki = 0.28 nM T98933 C1SM6H 44349600 Ki = 0.31 nM T98933 COFE32 44349601 Ki = 0.23 nM T98933 CB1P0S 44396251 Ki = 1900 nM T98933 CHY1C3 44396271 Ki > 2250 nM T98933 C29MBI 44396272 Ki > 2250 nM T98933 C4TQ6N 44396282 Ki = 1500 nM T98933 CH2Y3L 44396283 Ki > 2250 nM T98933 CWZB52 44396284 Ki > 2250 nM T98933 CD80LM 44396296 Ki > 2250 nM T98933 C6SI5L 44396297 Ki > 2250 nM T98933 CR4H1E 44396316 Ki > 2250 nM T98933 C45LRH 44396317 Ki > 2250 nM T98933 CA8V4G 44396331 Ki > 2250 nM T98933 CA8OB7 44400181 IC50 = 600 nM T98933 C4G9CF 44403605 IC50 = 2140 nM T98933 CW6EH8 44403606 IC50 = 9 nM T98933 C0L3WU 44403607 IC50 = 545 nM T98933 COU4B6 44403627 IC50 = 7.2 nM T98933 CVH75N 44403628 IC50 = 29 nM T98933 CTQ48J 44403634 IC50 = 0.3 nM T98933 C3SZ4I 44408427 IC50 = 15 nM T98933 CDE12F 44408544 EC50 = 4.3 nM T98933 C3TAU6 44408607 IC50 = 51 nM T98933 CM27EY 44417461 IC50 = 190 nM T98933 CC9BF0 44433089 IC50 = 26 nM T98933 C8QD9O 44434596 IC50 = 1.023 nM T98933 CLXF30 44434604 IC50 = 4.169 nM T98933 CP7C9J 44435761 IC50 = 100000 nM T98933 CWG53Q 44435778 IC50 = 33900 nM T98933 CH56GJ 44435779 IC50 = 43500 nM T98933 CB1UR7 44435786 IC50 = 69100 nM T98933 CL3FT4 44445692 IC50 = 3.467 nM T98933 C20LCQ 44445716 IC50 = 776.25 nM T98933 C1EGS9 44445719 IC50 = 190.55 nM T98933 CHT8I1 44445726 IC50 = 8.511 nM T98933 C9U7HY 44445727 IC50 = 870 nM T98933 C31JKD 44445730 IC50 = 9.55 nM T98933 C0NH4Z 44445731 IC50 = 239.88 nM T98933 CEX30A 44452442 EC50 = 58 nM T98933 CD38FN 44567764 EC50 = 70 nM T98933 CV1W9E 44589465 Ki = 31.3 nM T98933 C9K7HA 45270610 IC50 > 50000 nM T98933 CM7BY6 53385590 IC50 = 13000 nM T98933 C6Z7WI 60204885 EC50 = 550 nM T98933 C05ZRG 69428069 Ki = 14.1 nM T98933 CR2M8J 69844039 Ki = 31.7 nM T98933 C5SRF8 70681735 Ki = 20.3 nM T98933 C3A0DO 70682526 IC50 = 7400 nM T98933 CLJU20 70682537 IC50 = 2100 nM T98933 C2SVR8 70682538 IC50 = 2400 nM T98933 CBVQ29 70683842 Ki = 1.54 nM T98933 CVON79 70683843 Ki = 301 nM T98933 C9R0NB 70683844 Ki = 213 nM T98933 CG40IU 70684617 IC50 = 1700 nM T98933 CO1MQ8 70684618 IC50 = 2800 nM T98933 CU5VH3 70684619 IC50 = 8500 nM T98933 CARO49 70685018 Ki > 2250 nM T98933 CVK46F 70686763 IC50 = 8200 nM T98933 CWJ6U3 70686764 IC50 = 660 nM T98933 C70SIB 70688836 IC50 = 4200 nM T98933 CLF25D 70690926 IC50 = 5200 nM T98933 CB3ZC2 70690927 IC50 = 3400 nM T98933 C6FA0H 70690939 IC50 = 1400 nM T98933 C90XVL 70693065 IC50 = 1300 nM T98933 CC2EK8 70693080 IC50 = 1800 nM T98933 C2WC4V 70695111 IC50 = 7100 nM T98933 C92QMH 70695112 IC50 = 3300 nM T98933 CMNE57 70695113 IC50 = 310 nM T98933 CTQ37A 70697163 IC50 = 1600 nM T98933 CLU28H 71461159 EC50 = 0.47 nM T98933 CL8K9N 71523879 Ki = 1662 nM T98933 CQ0C5S 71523924 Ki = 441 nM T98933 C8DI5U 71523925 Ki = 124 nM T98933 CTU1K7 71523963 Ki = 223 nM T98933 CGHD73 71570928 IC50 = 16000 nM T98933 C49SBQ 71571065 IC50 = 5800 nM T98933 CE06XT 71571066 IC50 = 6600 nM T98933 CR92GT 71571067 IC50 = 3600 nM T98933 CTUC72 71571068 IC50 = 10600 nM T98933 C7UHM3 71571069 IC50 > 60000 nM T98933 C1P5HY 71571070 IC50 > 60000 nM T98933 C4CNP2 71571213 IC50 > 60000 nM T98933 CAV18D 71571215 IC50 > 60000 nM T98933 C97ISQ 71571216 IC50 = 20000 nM T98933 C5ZT9O 71716541 IC50 > 60000 nM T98933 C1TN8C 71716542 IC50 > 60000 nM T98933 CPJ4T2 71716543 IC50 > 60000 nM T98933 CP9B4C 71716544 IC50 > 60000 nM T98933 C4OE3H 71716545 IC50 > 60000 nM T98933 CIJ84X 71716546 IC50 = 59000 nM T98933 C4XL7Z 71716547 IC50 > 60000 nM T98933 C7BMG8 71716548 IC50 > 60000 nM T98933 C8O2NJ 71716549 IC50 > 60000 nM T98933 CA1Q0X 71716550 IC50 > 60000 nM T98933 CM6ZN5 71716551 IC50 > 60000 nM T98933 CX6RH7 71716552 IC50 > 60000 nM T98933 CTI7H2 71716553 IC50 > 60000 nM T98933 C8YEZ6 71716554 IC50 > 60000 nM T98933 CT3D1M 71717145 IC50 = 39000 nM T98933 CSHP85 71717146 IC50 > 60000 nM T98933 C5K3QG 71717147 IC50 > 60000 nM T98933 C6B5DO 71717148 IC50 > 60000 nM T98933 CK0ZQ9 71717149 IC50 > 60000 nM T98933 C96GSC 71717150 IC50 > 60000 nM T98933 C36SFW 71717155 IC50 > 60000 nM T98933 CLR58A 71717156 IC50 > 60000 nM T98933 CN4A9V 71717771 IC50 > 60000 nM T98933 CPLW58 71717772 IC50 > 60000 nM T98933 CIL03B 71717773 IC50 > 60000 nM T98933 C63QLG 71717774 IC50 = 38000 nM T98933 CV0I1H 71717775 IC50 > 60000 nM T98933 CUN4O0 71717776 IC50 > 60000 nM T98933 CSO2X5 71717777 IC50 > 60000 nM T98933 C52BZC 71717778 IC50 > 60000 nM T98933 CIE8V5 71717779 IC50 > 60000 nM T98933 C46ICD 71717780 IC50 > 60000 nM T98933 CPH02C 71718378 IC50 = 46000 nM T98933 COX71E 71718379 IC50 > 60000 nM T98933 CC94QZ 71718380 IC50 > 60000 nM T98933 CG2TH9 71718381 IC50 > 60000 nM T98933 C6G4BT 71718382 IC50 = 50000 nM T98933 CQ8AI1 71718383 IC50 > 60000 nM T98933 C4KOT9 71718386 IC50 > 60000 nM T98933 CH2TV1 71718387 IC50 > 60000 nM T98933 CXO1S7 71718388 IC50 > 60000 nM T98933 CI6AN0 71718985 IC50 = 24000 nM T98933 C5U7IR 71718986 IC50 > 60000 nM T98933 C0CJ8S 71718987 IC50 > 60000 nM T98933 C4KAZ7 71718988 IC50 > 60000 nM T98933 CIN3V1 71718992 IC50 > 60000 nM T98933 CZ3WG5 71718993 IC50 > 60000 nM T98933 CE6X2K 71718994 IC50 > 60000 nM T98933 C1IH2Q 71718995 IC50 > 60000 nM T98933 CN1RW4 71718996 IC50 > 60000 nM T98933 CKA36P 71718997 IC50 > 60000 nM T98933 C8LWP5 71719585 IC50 > 60000 nM T98933 CQ6BL0 71719586 IC50 > 60000 nM T98933 CFO1J2 71719587 IC50 > 60000 nM T98933 CT0DH9 71719588 IC50 > 60000 nM T98933 C3BT7V 71719589 IC50 > 60000 nM T98933 CBY36L 71719590 IC50 > 60000 nM T98933 C5SPB2 71719591 IC50 > 60000 nM T98933 CYNI30 71719592 IC50 > 60000 nM T98933 CJ5O6Q 71719593 IC50 > 60000 nM T98933 C7EKV1 71719594 IC50 > 60000 nM T98933 CB7O4D 71719597 IC50 > 60000 nM T98933 CD98PS 71719598 IC50 > 60000 nM T98933 CQ7U4O 71719599 IC50 > 60000 nM T98933 CXDE81 71719600 IC50 > 60000 nM T98933 CDM58X 71719601 IC50 > 60000 nM T98933 CCV8I1 71719602 IC50 > 60000 nM T98933 CH1EB5 71719603 IC50 > 60000 nM T98933 CX46KH 71719604 IC50 > 60000 nM T98933 C7KER0 71720182 IC50 > 60000 nM T98933 C0DYJ3 71720183 IC50 = 31000 nM T98933 CY4J2C 71720184 IC50 > 60000 nM T98933 C4Z0VS 71720185 IC50 > 60000 nM T98933 C5H0WP 71720186 IC50 > 60000 nM T98933 C9B4SP 71720187 IC50 > 60000 nM T98933 CHFZ51 71720188 IC50 > 60000 nM T98933 C2FM0U 71720189 IC50 > 60000 nM T98933 CUG52N 71720190 IC50 > 60000 nM T98933 CV1US9 71720192 IC50 > 60000 nM T98933 C7X8QB 71720193 IC50 > 60000 nM T98933 CB56IU 71720826 IC50 > 60000 nM T98933 CS5R7G 71720827 IC50 > 60000 nM T98933 CTF8D3 71720828 IC50 > 60000 nM T98933 CZ71PL 71720830 IC50 > 60000 nM T98933 C0Y9CT 71720831 IC50 > 60000 nM T98933 C5NU0T 71721539 IC50 > 100000 nM T98933 CP0G7O 73054742 EC50 = 150 nM T98933 CBJ8C9 73055020 EC50 = 37 nM T98933 CCO4X8 73055021 EC50 = 37 nM T98933 CZ8RJ5 73055022 EC50 = 62 nM T98933 C36LIJ 73055023 IC50 = 1100 nM T98933 C25DRF 73055024 IC50 = 1500 nM T98933 CANR79 76324858 IC50 = 24100 nM T98933 C4BA8W 90656430 IC50 > 69000 nM T98933 CO3KL0 118726602 Ki = 1.04 nM T98933 C45QSH 118726603 Ki = 1.12 nM T98933 CWQE31 118726604 Ki = 0.38 nM T98933 CZOI45 118726605 Ki = 0.26 nM T98933 C1QZ8J 118726606 Ki = 0.07 nM T98933 C0A9JB 118726607 Ki = 0.14 nM T98933 C94RVF 118726608 Ki = 0.04 nM T98933 C8IDF7 118726609 Ki = 0.18 nM T98933 C4KY2I 118726610 Ki = 0.09 nM T98933 CEW5K8 118726611 Ki = 0.3 nM T98933 CM2R8J 118726612 Ki = 0.54 nM T98933 CZM9O6 118726613 Ki = 0.64 nM T98933 CK8RB5 118726614 Ki = 1.11 nM T98933 CJA6K2 118726615 Ki = 3.14 nM T98933 C2J8PF 118726616 Ki = 8.04 nM T98933 CH1FA8 135528521 IC50 = 22 nM T98933 C0FWQ7 135559141 IC50 = 138.04 nM T98933 CU20KW 135559142 IC50 = 123.03 nM T98933 CW9R4B 135559143 IC50 = 28.18 nM T98933 CCF02H 145964530 IC50 = 7600 nM T98933 C56SHA 145964597 IC50 = 8800 nM T98933 C5H8EZ 145965425 IC50 = 970 nM T98933 C98CHS 145977976 IC50 = 9800 nM T98933 D01HAZ 23635364 IC50 = 4200 nM T98933 D01NTN 11350323 IC50 = 360 nM T98933 D01WVE 9872203 IC50 = 4100 nM T98933 D02CGG 44435789 IC50 = 8200 nM T98933 D03VOM 3092218 IC50 = 4300 nM T98933 D03XCG 23635367 IC50 = 15200 nM T98933 D05FRX 11153607 IC50 = 800 nM T98933 D05XMM 44186304 IC50 = 8100 nM T98933 D05ZJC 9925361 IC50 = 1905.46 nM T98933 D06IJW 23635362 IC50 = 2700 nM T98933 D07MAF 21653696 IC50 = 9600 nM T98933 D08BQI 11291923 IC50 = 5700 nM T98933 D09XOC 23635858 IC50 = 3000 nM T98933 D0A5XG 10027822 IC50 = 370 nM T98933 D0G7HF 23635860 IC50 = 19100 nM T98933 D0H6BV 24843916 IC50 = 4100 nM T98933 D0I2GK 71212 EC50 = 3.5 nM T98933 D0I7DH 23635476 IC50 = 7600 nM T98933 D0J0MD 23635730 IC50 = 17900 nM T98933 D0Q9ZN 23648092 IC50 = 230 nM T98933 D0U0GY 44435784 IC50 = 10500 nM T98933 D0U9JC 44435785 IC50 = 11400 nM T98933 D0YU9Z 14899645 IC50 = 18600 nM T98933 D0ZX0Y 23635856 IC50 = 6200 nM T39996 D02HFD 124886 IC50 > 100000 nM T39996 D07BDD 65359 IC50 > 100000 nM T39996 D0V0LB 6058 IC50 > 100000 nM T39996 D0X5SD 3117 IC50 = 1600 nM T39996 D0B1FE 3194 IC50 = 730 nM T39996 D09YFD 21928 IC50 = 1100 nM T39996 D0X2AU 23427 IC50 = 4900 nM T39996 CF3N7H 5941 IC50 > 100000 nM T39996 C8IWZ0 10236 IC50 > 100000 nM T39996 CGJ83B 15460 IC50 = 860 nM T39996 CX1LG8 65093 IC50 = 2700 nM T39996 C95WZA 123446 IC50 = 1500 nM T39996 CJ7FR6 533728 IC50 = 81000 nM T39996 C37UOC 590397 IC50 = 1000 nM T39996 CQE8T5 5462814 IC50 = 1700 nM T39996 C85NAQ 24858111 IC50 = 65000 nM T39996 C5N3LG 44251522 IC50 = 58 nM T39996 CCI45D 44604812 IC50 = 4 nM T39996 CFU9H7 44605025 IC50 = 12 nM T39996 CL76QF 44605026 IC50 = 13 nM T39996 CFQ17S 44605027 IC50 = 23 nM T39996 C6PY2V 44605028 IC50 = 11 nM T39996 CZF8V7 46174173 IC50 = 100 nM T39996 C70VHB 53315882 IC50 < 15 nM T39996 C7M0FJ 59457983 IC50 = 600000 nM T39996 CAVD69 70678415 IC50 = 25000 nM T39996 C52YJT 76310995 IC50 = 100000 nM T39996 CNQ86R 76314627 IC50 = 500000 nM T39996 CYB1U4 76318201 IC50 = 100000 nM T39996 CZ09ML 76321898 IC50 = 400000 nM T39996 C4XJ5N 78357767 IC50 > 100000 nM T39996 CCT09O 86288827 IC50 = 87000 nM T39996 C01DAP 86288828 IC50 = 1500 nM T39996 CA18TS 90655765 IC50 = 235000 nM T39996 C5NX4U 90655766 IC50 = 147000 nM T39996 C9BI8F 118607414 IC50 = 180 nM T39996 C7X2AQ 118613624 IC50 > 20000 nM T39996 C7TI9A 129012136 IC50 = 5 nM T39996 C6F2VK 129012137 IC50 = 4 nM T39996 CJI14M 129072680 IC50 > 20000 nM T39996 COL81P 129085358 IC50 > 20000 nM T39996 CTQE45 132471834 IC50 = 18 nM T39996 CBO31X 132471835 IC50 = 6 nM T39996 CL2ZI0 132609264 IC50 = 794300 nM T39996 CYJR92 132609265 IC50 = 21800 nM T39996 CBTH20 137348638 IC50 = 7 nM T39996 CR53YC 137631913 IC50 = 6 nM T39996 C8VT5L 137632046 IC50 = 203700 nM T39996 C8VO5D 137632076 IC50 = 44 nM T39996 C5AC6M 137632524 IC50 = 20 nM T39996 C46WLE 137633319 IC50 > 5000 nM T39996 CIB30Q 137633627 IC50 = 34 nM T39996 C8AM9L 137635489 IC50 = 808 nM T39996 CE60DR 137635748 IC50 = 12 nM T39996 CTU4G0 137636690 IC50 = 20 nM T39996 CI5Q3X 137636915 IC50 = 26 nM T39996 CK1WU6 137637870 IC50 = 28 nM T39996 C3TD2E 137638286 IC50 = 15 nM T39996 CO6JA8 137639333 IC50 > 5000 nM T39996 CO78IY 137639766 IC50 = 73 nM T39996 C0EYN9 137639969 IC50 = 20 nM T39996 CCSI40 137640754 IC50 = 17 nM T39996 C2P3JR 137640823 IC50 = 47700 nM T39996 C5TY4L 137640829 IC50 = 159 nM T39996 C7G9AB 137643064 IC50 = 46 nM T39996 CV4PI3 137643498 IC50 > 6000 nM T39996 C2DWX9 137643972 IC50 = 95100 nM T39996 CZM39K 137644029 IC50 = 1230 nM T39996 CS9RO5 137644870 IC50 = 11 nM T39996 C6NW5B 137645215 IC50 = 59 nM T39996 C6WLD1 137645686 IC50 = 11 nM T39996 CZTV84 137646234 IC50 = 18 nM T39996 C9EP0L 137647456 IC50 = 58 nM T39996 CN5UY2 137647689 IC50 > 1000 nM T39996 CD2JQ9 137648196 IC50 = 77 nM T39996 C7Y2RH 137648735 IC50 = 115000 nM T39996 CJO19V 137649514 IC50 = 135 nM T39996 CZD47A 137649599 IC50 = 35 nM T39996 CZR86C 137650174 IC50 = 24 nM T39996 CUM43J 137650973 IC50 = 145800 nM T39996 CSU4J8 137651295 IC50 = 97 nM T39996 CJ57XR 137652778 IC50 = 29 nM T39996 C8N2BU 137653025 IC50 = 12 nM T39996 C4JYZ0 137654123 IC50 = 341 nM T39996 CES2Y4 137654330 IC50 = 50 nM T39996 CF65YG 137654447 IC50 = 18 nM T39996 CX2RM3 137654889 IC50 = 43 nM T39996 C8MQ2I 137655652 IC50 = 24 nM T39996 C3BI4K 137655660 IC50 = 35 nM T39996 CHS71L 137656981 IC50 = 23 nM T39996 CYF6V9 137657228 IC50 = 27 nM T39996 C0R6QN 137658284 IC50 = 63 nM T39996 CR7GF2 137658708 IC50 = 16 nM T39996 CDQW60 137661215 IC50 > 5000 nM T39996 C19VQE 137661488 IC50 = 36 nM T39996 CD1K7J 137661663 IC50 = 28 nM T39996 C85XIG 137662224 IC50 = 30 nM T39996 C8LEV4 139267760 IC50 > 10000 nM T39996 CJT6G1 155511077 IC50 = 19 nM T39996 C4NS2X 155512777 IC50 = 18500 nM T39996 CO5P4T 155513225 IC50 = 41 nM T39996 CDWR24 155515450 IC50 = 10300 nM T39996 C04DFY 155516671 IC50 = 1460 nM T39996 CB9WP0 155517958 IC50 = 179 nM T39996 CFLK08 155520544 IC50 = 300 nM T39996 CYOD10 155522526 IC50 = 1080 nM T39996 CJOW75 155522891 IC50 = 19 nM T39996 CL4T2Q 155523641 IC50 = 280 nM T39996 CCI9U8 155524518 IC50 = 926 nM T39996 C4UXQ1 155526805 IC50 = 3090 nM T39996 CLQ18S 155527069 IC50 = 4090 nM T39996 CP60DZ 155527429 IC50 = 698 nM T39996 CG2EM1 155527465 IC50 = 53600 nM T39996 CH5X4E 155527661 IC50 = 16 nM T39996 CD8C5B 155528012 IC50 = 44 nM T39996 CKN4C6 155528155 IC50 = 9 nM T39996 C53YIH 155530887 IC50 = 12 nM T39996 CA9P6Y 155532307 IC50 = 9 nM T39996 C1J5TI 155532811 IC50 = 2860 nM T39996 CI0ML6 155534407 IC50 = 1350 nM T39996 C6FEP9 155535898 IC50 = 679 nM T39996 CU2XG3 155537180 IC50 = 953 nM T39996 C7Q9HD 155537279 IC50 = 47 nM T39996 C6R7JS 155537616 IC50 = 78 nM T39996 C78EAT 155538085 IC50 = 70 nM T39996 C5NH2I 155540357 IC50 = 1950 nM T39996 C9H4GL 155540760 IC50 = 205 nM T39996 C5OGN0 155542626 IC50 = 642 nM T39996 CHL9F7 155543202 IC50 = 1550 nM T39996 CT3M4J 155543558 IC50 = 1250 nM T39996 CQ20HW 155544061 IC50 = 3470 nM T39996 C0VJO4 155545582 IC50 = 2470 nM T39996 C2I8ES 155546390 IC50 = 529 nM T39996 CBLI45 155547053 IC50 = 2650 nM T39996 C51VKD 155547438 IC50 = 12 nM T39996 C8RD2L 155548665 IC50 = 4670 nM T39996 C8Q3GX 155550036 IC50 = 885 nM T39996 CSKE02 155550699 IC50 = 1310 nM T39996 C1QOP9 155550708 IC50 = 11 nM T39996 CS1TK5 155551475 IC50 = 2360 nM T39996 CJAT69 155553711 IC50 = 3990 nM T39996 CTIM98 155556005 IC50 = 27 nM T39996 CV9EZ2 155556376 IC50 = 2010 nM T39996 CVT50L 155557402 IC50 = 35 nM T39996 CYAP13 155557747 IC50 = 122 nM T39996 C5KZP1 155558337 IC50 = 19 nM T39996 CQ08KG 155559900 IC50 = 94 nM T39996 C2FIO6 155559947 IC50 = 2230 nM T39996 CD3HO4 155562561 IC50 = 7510 nM T39996 C0J6AT 155562781 IC50 = 152 nM T39996 C91BWQ 155564365 IC50 = 2380 nM T39996 C5VN8K 155564441 IC50 = 647 nM T39996 CVZ2C4 155565339 IC50 = 150 nM T39996 C84AKC 155566143 IC50 = 6 nM T39996 D00FLT 65482 IC50 = 100 nM T39996 D02UVS 5455 IC50 = 1100 nM T39996 D06PPL 25150857 IC50 = 700 nM T39996 D09CLP 439155 IC50 = 230 nM T39996 D0BI4T 53315878 IC50 < 2.5 nM T39996 D0C5EG 76285486 IC50 = 11 nM T39996 D0CX4W 46901937 IC50 = 15 nM T39996 D0DQ6Z 8530 IC50 = 14000 nM T39996 D0GK7A 46224516 IC50 = 19 nM T39996 D0L5LN 6780 IC50 > 100000 nM T39996 D0RO9T 73755260 IC50 = 1600 nM T54128 D00ENY 33032 IC50 = 613 nM T54128 D02VKC 3272524 Ki = 70 nM T54128 D0B0NQ 127894 IC50 = 1350 nM T54128 D02QZL 9903685 IC50 = 80 nM T54128 D06WHL 135484540 IC50 = 700 nM T54128 D0H1FV 68736 IC50 = 967 nM T54128 CO3XI2 125406 IC50 = 88000 nM T54128 C6RD3L 125407 IC50 = 12000 nM T54128 C32DCS 3018579 IC50 = 6700 nM T54128 C5OHM8 3481675 IC50 = 30 nM T54128 CRL5Z4 5353536 IC50 = 340 nM T54128 CS5V4U 5486548 Ki = 135 nM T54128 CB50FH 6604872 IC50 = 3000 nM T54128 C20IEF 9837860 IC50 = 5700 nM T54128 CW79HF 9909062 Ki = 215 nM T54128 C4SG1T 9927756 Ki = 600 nM T54128 CI7GM6 9937279 Ki = 7 nM T54128 CHIL12 9985663 Ki = 4 nM T54128 CPF74Y 10017901 IC50 = 153 nM T54128 CM5I3E 10036285 IC50 = 24000 nM T54128 C4LWR8 10037930 IC50 = 7000 nM T54128 CB8KW6 10048025 IC50 = 340 nM T54128 C76YSF 10051732 Ki = 15 nM T54128 C5G2WD 10084218 IC50 = 84500 nM T54128 C6XJD8 10244065 IC50 = 8000 nM T54128 C5NOI8 10244106 IC50 > 100000 nM T54128 C0AC4T 10247474 Ki = 180 nM T54128 C8THG7 10266209 IC50 = 166 nM T54128 C70WBQ 10401891 IC50 = 44000 nM T54128 CX1V3L 10437436 Ki = 5 nM T54128 C5M4IH 10538709 IC50 > 100000 nM T54128 CYX93H 10562939 IC50 = 94 nM T54128 C7WKJ2 10610792 IC50 > 100000 nM T54128 C6A1UE 10656900 IC50 > 100000 nM T54128 C0O6ZI 10658567 IC50 = 54000 nM T54128 C9BV5R 10729534 IC50 = 5800 nM T54128 CIW54Y 10752476 IC50 = 1500 nM T54128 C9H0TI 10800053 IC50 = 72000 nM T54128 C3B9HI 10823814 IC50 = 48000 nM T54128 C02QUD 10824747 IC50 = 700 nM T54128 CXLW54 11948707 Ki > 10000 nM T54128 CJZ6K9 15337998 Ki = 1500 nM T54128 CZ8BM3 15840183 Ki = 450 nM T54128 CT4ZO6 15840184 Ki = 54 nM T54128 C06MHR 15840185 Ki = 4 nM T54128 C3A5ES 15840186 Ki = 4 nM T54128 C1QA4W 15840187 Ki = 20 nM T54128 CT1I3Y 21710164 Ki = 10000 nM T54128 CB9E5R 21710166 Ki = 980 nM T54128 CL3UT2 22097086 Ki = 3000 nM T54128 CLRK62 22097088 Ki = 70 nM T54128 CJ52FG 22097105 Ki = 400 nM T54128 C4J3TO 22097119 Ki = 78 nM T54128 CD7H5E 22097148 Ki = 20000 nM T54128 C62FHX 22097151 Ki = 2000 nM T54128 CR5BZ4 22097158 Ki > 25000 nM T54128 CE20FP 22097165 Ki = 210 nM T54128 C3BKT5 22097178 Ki = 76 nM T54128 C72VRZ 22097186 Ki > 25000 nM T54128 CVD94P 22097194 Ki = 250 nM T54128 C9EO8L 22097211 Ki > 25000 nM T54128 C2H4CP 22100063 Ki = 95 nM T54128 C76PHV 22100072 Ki = 110 nM T54128 CM2H1L 22100104 Ki = 2000 nM T54128 CCMS36 22100119 Ki = 49 nM T54128 C1DMH8 22100133 Ki = 5 nM T54128 CJ8UB0 22100152 Ki = 840 nM T54128 CLX8S4 22100157 Ki = 71 nM T54128 CIG65E 22449297 Ki = 22 nM T54128 CM2AN8 44268202 Ki = 250 nM T54128 C5ES0F 44268209 Ki = 880 nM T54128 C9WG8T 44268224 Ki = 280 nM T54128 CG09WU 44268242 Ki = 500 nM T54128 CL0H9R 44268310 Ki = 3000 nM T54128 CJUL-93 44268318 Ki = 650 nM T54128 C49GIP 44268353 Ki = 140 nM T54128 C8V4DX 44268357 Ki = 890 nM T54128 CMC3B8 44268369 Ki > 25000 nM T54128 CRUJ15 44281577 IC50 = 1350 nM T54128 C4ZX5R 44281591 IC50 = 630 nM T54128 CT1X5A 44281631 IC50 = 580 nM T54128 C8GQ4A 44304811 IC50 = 1350 nM T54128 CWAX82 44317999 Ki = 60 nM T54128 C9J4ME 44348419 IC50 = 4300 nM T54128 C1JRT2 44377742 IC50 = 21000 nM T54128 C3YN8I 44377743 IC50 = 36000 nM T54128 C6PYE7 44379376 IC50 = 14000 nM T54128 CGX3P0 44460610 Ki = 66 nM T54128 CDI84E 71450922 IC50 > 10000 nM T54128 CDA4O8 135407136 IC50 = 2100 nM T54128 C0TK2B 135453826 IC50 = 1900 nM T54128 C4E0VH 135484474 IC50 = 150 nM T54128 C1ET2K 135535891 IC50 = 1800 nM T54128 CR45DZ 135976300 IC50 = 7200 nM T54128 CP9TR0 10324985 Ki > 10000 nM T54128 D03RGP 1221 IC50 = 23 nM T54128 D04DHB 1779 IC50 > 100000 nM T54128 D05KQC 3899541 IC50 = 200 nM T54128 D0J3EZ 4038142 IC50 = 2000 nM T54128 D0S6TW 1845 IC50 = 27000 nM T82739 D05PHH 3447 IC50 = 1350 nM T82739 D0I0RJ 16231 IC50 > 50000 nM T82739 D0ID3W 9911502 IC50 = 15800 nM T82739 D0PK7J 56599309 Ki = 2.4 nM T82739 D0D5RH 11641515 IC50 = 12000 nM T82739 D0N7WR 108040 Ki = 570 nM T82739 C1BHS3 193409 Ki = 22500 nM T82739 CR4KE5 445844 Ki = 800 nM T82739 C87OTC 447733 Ki = 7170 nM T82739 CF6D4B 447734 Ki = 2720 nM T82739 CHT05K 447735 Ki = 436 nM T82739 CCKZ79 668744 IC50 = 30100 nM T82739 C53FNM 674593 IC50 = 11900 nM T82739 C45NBS 674629 IC50 = 4400 nM T82739 C21HDC 674632 IC50 = 11300 nM T82739 CBX3U0 674652 IC50 = 6600 nM T82739 C98EGA 741761 IC50 > 50000 nM T82739 CFD4M6 747662 IC50 > 50000 nM T82739 C9D4IN 754821 IC50 > 50000 nM T82739 C0ER8S 767161 IC50 = 60500 nM T82739 CLR3H1 899247 IC50 = 42200 nM T82739 CQ2R0M 1011274 IC50 = 28100 nM T82739 C7P1UO 1201257 IC50 = 31700 nM T82739 C2PRY6 1269450 IC50 = 67400 nM T82739 CO4AB7 2264784 IC50 = 5500 nM T82739 CTE79D 3011892 Ki > 50000 nM T82739 CU43OY 3088969 Ki > 50000 nM T82739 C0K7TF 3123858 IC50 > 50000 nM T82739 C8KD9E 3162843 IC50 > 50000 nM T82739 CQY92E 3660962 IC50 = 7200 nM T82739 CQWL43 5039074 IC50 = 35400 nM T82739 CLD0C6 5348879 IC50 = 96200 nM T82739 C1B9GP 5400404 IC50 > 50000 nM T82739 CF1P5H 5430316 IC50 = 54200 nM T82739 CZ1XU5 5876194 IC50 = 13500 nM T82739 CG2A7X 7028541 IC50 = 120100 nM T82739 C6JDM9 9799627 Ki = 145 nM T82739 C2F5NS 9884570 Ki = 110 nM T82739 CKDP84 9895193 Ki = 7200 nM T82739 C0LKE7 9912771 Ki = 11000 nM T82739 CC0D5H 9915041 Ki = 58 nM T82739 CH8QJ4 9916876 IC50 = 14 nM T82739 CF9SD1 9917846 IC50 = 29 nM T82739 C8F5CW 9937921 Ki = 61 nM T82739 CNE34O 9939021 IC50 = 120 nM T82739 CX85LD 9954980 Ki > 16000 nM T82739 CM7IF6 9956559 Ki > 20000 nM T82739 CBC2K3 9959749 IC50 = 130 nM T82739 CA9S3O 9981709 IC50 = 41000 nM T82739 C7BD9S 10024676 IC50 = 19000 nM T82739 C7LZ2T 10050676 IC50 = 25000 nM T82739 CQP65H 10095093 Ki = 19000 nM T82739 C3OG5U 10095865 IC50 = 5010 nM T82739 C1VT4F 10117027 Ki = 3000 nM T82739 C31QAL 10143532 Ki > 2300 nM T82739 C5I0YH 10168444 Ki = 17000 nM T82739 CSVF04 10253001 IC50 = 28000 nM T82739 CQ9ZO1 10275412 Ki = 8900 nM T82739 CP64HV 10342843 Ki > 1000000 nM T82739 CK9J7X 10343728 IC50 = 25100 nM T82739 C6JF0P 10365153 IC50 = 35000 nM T82739 C10ISY 10367012 Ki = 5000 nM T82739 C57GFJ 10386993 IC50 = 16000 nM T82739 C6S4CO 10391715 Ki = 14000 nM T82739 CT75ZJ 10411941 IC50 = 16000 nM T82739 CBV6N7 10423722 IC50 > 50000 nM T82739 CJTH60 10432907 Ki = 3330 nM T82739 C6AZ8B 10435038 Ki = 8600 nM T82739 CISN08 10455169 IC50 = 54000 nM T82739 C6KJM2 10461790 Ki > 50000 nM T82739 CV0X6G 10480463 IC50 = 560 nM T82739 CEI65Z 10483775 Ki = 4.6 nM T82739 C5ED3G 10529121 Ki = 79000 nM T82739 CU8N3V 10578280 Ki = 7300 nM T82739 C8SUZ9 10624948 Ki = 12000 nM T82739 CEJ14F 10624997 Ki = 3300 nM T82739 CR5EX8 10648196 Ki = 7600 nM T82739 CPWH69 10648370 Ki = 35000 nM T82739 CJG9H6 10669349 Ki = 586000 nM T82739 C5VB1U 10695159 Ki = 18000 nM T82739 CP4QC5 10696511 Ki = 775000 nM T82739 CGYR23 10696955 Ki = 15000 nM T82739 CPGV87 10718240 Ki = 36000 nM T82739 CIKF89 10719580 Ki = 170000 nM T82739 CZ0Q8K 10742217 Ki = 816000 nM T82739 C7RWD8 10744643 Ki = 399000 nM T82739 CKOQ35 10767421 Ki = 29000 nM T82739 C3IN8W 10815545 Ki = 27000 nM T82739 CVQE76 10816339 Ki = 58000 nM T82739 CLB15C 10871563 Ki = 4800 nM T82739 C2TBO9 10959252 Ki = 600 nM T82739 CAD15G 11149953 Ki = 8000 nM T82739 C6LVG4 11186243 Ki = 2570 nM T82739 CTX9F3 11188793 Ki = 1350 nM T82739 CLA93S 11237163 Ki = 8458 nM T82739 CHLK70 11244460 Ki = 2430 nM T82739 C86DZB 11292119 Ki = 230 nM T82739 C6CDN3 11347670 Ki = 18100 nM T82739 CLY5G8 11350400 Ki = 849 nM T82739 CR8NW9 11351302 Ki > 10000 nM T82739 CTJ1Z2 11361949 Ki = 400 nM T82739 C63LIR 11473486 Ki = 1370 nM T82739 CK34OX 11509611 Ki = 330 nM T82739 CO68MA 11524737 Ki = 940 nM T82739 CJP9O1 11684611 Ki = 5 nM T82739 CQ5U8H 11739438 Ki = 112 nM T82739 C7WJP0 11754749 IC50 = 26000 nM T82739 C7JLR1 11774107 Ki = 4300 nM T82739 CNO67W 11798089 Ki = 14000 nM T82739 CYX74A 11824584 Ki = 1300 nM T82739 C2QO1B 15955412 Ki > 50000 nM T82739 C19ARJ 15984063 Ki = 43000 nM T82739 C53YRO 16098910 IC50 = 10 nM T82739 CN6CJ2 16220264 IC50 = 1340 nM T82739 CJSL38 18727836 IC50 = 300 nM T82739 CRX19I 23646295 Ki > 2300 nM T82739 CKH4O5 24180463 Ki > 6000 nM T82739 C7WTO3 24689997 IC50 = 8600 nM T82739 CTE3P4 24692287 IC50 = 20600 nM T82739 CJUE04 24860432 IC50 > 50000 nM T82739 C0UA9T 24860449 IC50 > 50000 nM T82739 C52CJA 24860451 IC50 > 50000 nM T82739 CZI85G 24984725 Ki = 0.1 nM T82739 CN0ZW3 24999867 Ki > 1000 nM T82739 CEM32W 25001205 Ki > 1000 nM T82739 C4Q9XM 25166807 Ki = 130 nM T82739 CX6A4M 25166808 Ki = 170 nM T82739 C2H4PJ 25166809 Ki = 122 nM T82739 CF1I6Q 25166810 Ki = 270 nM T82739 C9W0GO 25167018 Ki = 120 nM T82739 CHB21I 44265055 IC50 = 12000 nM T82739 CNK8W1 44310877 IC50 = 710 nM T82739 C8KOM9 44333945 Ki = 15500 nM T82739 CH32DA 44333955 Ki = 28 nM T82739 C75KOP 44333957 Ki = 500 nM T82739 C7A6KF 44333986 Ki = 4 nM T82739 CF1LQ4 44333999 Ki = 89 nM T82739 CZ7RK3 44334001 Ki = 5 nM T82739 CUO4N2 44334160 Ki = 2 nM T82739 CRT4G3 44335601 Ki = 22000 nM T82739 C7Z9WL 44335624 Ki = 97000 nM T82739 CAY34C 44347478 Ki > 1000000 nM T82739 CT0QN1 44347480 Ki = 476000 nM T82739 C1UN9I 44347534 Ki = 767000 nM T82739 C0V2FL 44347624 Ki = 1000000 nM T82739 CZ8XL6 44385679 IC50 = 210 nM T82739 CL5BA4 44385729 IC50 = 640 nM T82739 C3D2CL 44385935 IC50 = 500 nM T82739 CW08OY 44385998 IC50 = 790 nM T82739 CV6KG4 44386059 IC50 = 380 nM T82739 C5MR1F 44386934 IC50 = 500 nM T82739 C78QJO 44394249 Ki > 50000 nM T82739 CQRB69 44394250 Ki > 50000 nM T82739 CTS5W9 44404049 IC50 > 400000 nM T82739 C3BX5Y 44412781 Ki = 83000 nM T82739 CIP7E1 44415075 IC50 = 46200 nM T82739 C0THI1 44415189 IC50 = 75000 nM T82739 CVO5Q1 44432538 Ki > 10000 nM T82739 CR16BF 44434808 Ki > 10800 nM T82739 CQIX73 44434809 Ki > 6000 nM T82739 COG34X 44434818 Ki > 6000 nM T82739 C9T1DP 44434835 Ki > 10800 nM T82739 CB86HU 44453827 IC50 = 13 nM T82739 CVZW52 44537923 IC50 = 19000 nM T82739 COX6G5 52943174 IC50 = 1.7 nM T82739 CDH59M 52944043 IC50 = 2000 nM T82739 C8VI6M 52944358 IC50 = 39.1 nM T82739 CNA7U8 52946795 IC50 = 1500 nM T82739 C0T3CX 52948030 IC50 > 10000 nM T82739 CA6GQ5 53341037 Ki = 70 nM T82739 CIKQ81 53345652 Ki = 1.5 nM T82739 CXWS90 53345968 Ki = 0.3 nM T82739 C76GSI 53346181 Ki = 7.5 nM T82739 CV60BK 53488415 Ki = 6218 nM T82739 CI2ND0 54741583 Ki = 28 nM T82739 C17MSO 56640092 Ki = 136 nM T82739 CGP7Y6 56640160 Ki = 25.3 nM T82739 C30AJK 56640226 Ki = 19 nM T82739 CH1EI8 56954620 Ki = 25.4 nM T82739 C4EHU8 56954732 Ki = 868 nM T82739 C5C8XO 56954733 Ki = 493 nM T82739 CST4F0 56954834 Ki = 17.4 nM T82739 CRK92A 56954952 Ki = 10.1 nM T82739 CLY4C9 57390236 IC50 = 910000 nM T82739 CPBW48 57392333 Ki = 2000000 nM T82739 CEO1L3 57393799 IC50 = 380000 nM T82739 CL2JE5 57395841 Ki = 3300000 nM T82739 CXZ3D0 57400764 IC50 = 680000 nM T82739 CMG29L 57404341 IC50 = 1700 nM T82739 CXGW36 57404342 IC50 = 300 nM T82739 CTE30K 57842560 Ki > 6000 nM T82739 C0C6UB 57842624 Ki = 3600 nM T82739 C7XY5A 57842673 Ki > 6000 nM T82739 C41NSR 57842812 Ki = 50 nM T82739 C9XW1C 57842830 Ki > 10000 nM T82739 CWF0C3 57842850 Ki = 4600 nM T82739 C73CPB 57842913 Ki = 1700 nM T82739 C60HCV 57976401 Ki = 519 nM T82739 CHB27Y 57976410 Ki = 1850 nM T82739 CM8UJ7 57976444 Ki = 41 nM T82739 CQ71KE 57976446 Ki = 240 nM T82739 CSC0L5 59020200 Ki > 11000 nM T82739 CPW2H7 59315536 Ki > 10000 nM T82739 CL42XV 59401924 Ki = 350 nM T82739 CHJI56 59401943 Ki = 24 nM T82739 CA76HG 59401978 Ki = 340 nM T82739 CO38AC 59402011 Ki = 110 nM T82739 CVG75I 59402039 Ki = 23 nM T82739 CF26ZO 59402046 Ki > 6000 nM T82739 C7IWJ3 59402077 Ki = 20 nM T82739 CTW85S 59402125 Ki = 240 nM T82739 CKX9B7 59402220 Ki = 46 nM T82739 CZD0N4 59402226 Ki > 6000 nM T82739 CK7I1A 59402239 Ki = 210 nM T82739 C6JP8Q 60154989 Ki = 2 nM T82739 CE5A7B 60162406 Ki = 320 nM T82739 C3LT2W 66674079 Ki = 3820 nM T82739 CYH7X1 66674212 Ki = 3440 nM T82739 C3ND0L 66674351 Ki = 2217 nM T82739 C5N1GU 66674475 Ki = 4500 nM T82739 C23QOJ 66674821 Ki = 1924 nM T82739 CWOD93 66744646 Ki = 16 nM T82739 CKWQ82 67155200 Ki = 2900 nM T82739 C0SDB3 68020667 Ki = 392 nM T82739 C17JAZ 68284084 IC50 > 30000 nM T82739 C6AU1R 70252985 Ki = 268 nM T82739 CTO5I6 70253788 Ki = 1370 nM T82739 C8A7ZJ 70306716 Ki = 0.019 nM T82739 C1A2FN 70681010 IC50 = 13500 nM T82739 CHC3B5 70683145 IC50 = 12900 nM T82739 CM5BH2 70683146 IC50 = 3800 nM T82739 C4IFW3 70683249 Ki = 0.075 nM T82739 CN38UY 70687492 Ki = 9.4 nM T82739 C3Z7RM 70695744 IC50 = 7800 nM T82739 CC2Q7G 70695750 IC50 = 10600 nM T82739 CJPF90 71548883 Ki = 310 nM T82739 C30ZKJ 71561420 Ki = 1000 nM T82739 CH32TL 71561557 Ki = 187 nM T82739 C8RW7E 71562631 Ki = 3.2 nM T82739 C4UHB2 71562760 Ki = 118 nM T82739 C0EM6D 71562761 Ki = 24 nM T82739 CNS21T 71562882 Ki = 240 nM T82739 C3SBE2 71562883 Ki = 422 nM T82739 C2NY0B 71563006 Ki = 500 nM T82739 CG46AZ 71563007 Ki = 242 nM T82739 C2O4SB 71563124 Ki = 440 nM T82739 C4CT8O 71563125 Ki = 116 nM T82739 C78DJQ 71711730 IC50 < 10000 nM T82739 CS2CR9 71716063 IC50 = 20 nM T82739 C45APQ 71716064 IC50 = 30 nM T82739 C64YFO 71716065 IC50 = 50 nM T82739 CD53RA 71716975 Ki = 0.3 nM T82739 CSP5T2 71716976 Ki > 120000 nM T82739 CAR2J6 71717264 IC50 = 28.6 nM T82739 CWJ75U 71717265 IC50 = 30 nM T82739 C7JDE3 71719101 IC50 = 800 nM T82739 CQ3K2V 71719191 Ki = 12.9 nM T82739 C1Y0JV 71719710 IC50 = 21.2 nM T82739 C24UEO 71720319 IC50 = 1800 nM T82739 CVCM38 71818688 IC50 = 11200 nM T82739 CLI36U 72551247 Ki = 520 nM T82739 C01LOR 73051877 Ki = 3 nM T82739 C6M9ZP 73052197 Ki = 9 nM T82739 CXJ86Q 73052510 Ki = 1 nM T82739 CB14LR 73052831 Ki = 2.39 nM T82739 CU9C2F 73345352 IC50 = 7181 nM T82739 CDQP51 73347119 Ki > 50000 nM T82739 CM3PH8 73350210 Ki > 50000 nM T82739 C9ASZ2 86302628 IC50 > 1000000 nM T82739 CMD5V7 86583041 Ki = 24 nM T82739 CO6U9I 88582319 Ki > 6000 nM T82739 C9A7YX 90655485 IC50 > 1000000 nM T82739 C90UNY 90655486 IC50 = 740000 nM T82739 C75WHK 90655487 IC50 > 1000000 nM T82739 CZ1Q2P 90655488 IC50 > 1000000 nM T82739 CSG0L5 90655489 IC50 > 1000000 nM T82739 C8KX5F 90655490 IC50 > 1000000 nM T82739 C9W1CO 90655491 IC50 > 1000000 nM T82739 C5WIF7 90655492 IC50 > 1000000 nM T82739 C6FE2K 90655493 IC50 > 1000000 nM T82739 C2I7SQ 90655494 IC50 > 1000000 nM T82739 CXY0I6 90655495 IC50 > 1000000 nM T82739 CWL8U1 90655496 IC50 > 1000000 nM T82739 CRQ6I4 90655497 IC50 > 1000000 nM T82739 CL27GQ 90655498 IC50 > 1000000 nM T82739 CLG8M0 90655499 IC50 > 1000000 nM T82739 CBK7Y9 90655500 IC50 > 1000000 nM T82739 CD7WM6 90655501 IC50 > 1000000 nM T82739 CJ7B8Y 90655502 IC50 > 1000000 nM T82739 CW6VS9 90655503 IC50 > 1000000 nM T82739 CV1NM4 90655504 IC50 > 1000000 nM T82739 CKPN23 90655505 IC50 > 1000000 nM T82739 CZ8S4C 90655506 IC50 > 1000000 nM T82739 C65TLW 101862198 Ki > 1000000 nM T82739 CI4KC5 117986603 IC50 = 7.2 nM T82739 C3MVG0 118720988 Ki = 1360 nM T82739 C9M2IH 118720990 Ki = 1170 nM T82739 C1E6GW 118720991 Ki = 1470 nM T82739 C9BVI5 118720993 Ki = 5540 nM T82739 C1FQZ6 118720994 Ki = 60 nM T82739 C0WZA2 118720996 Ki = 220 nM T82739 CE89KB 118720997 Ki = 5270 nM T82739 CIAL50 118720998 Ki = 765 nM T82739 C4HLM3 118720999 Ki = 1310 nM T82739 CLD6I3 118721000 Ki = 910 nM T82739 C0XG7H 118721001 Ki = 920 nM T82739 CZC53M 118721002 Ki = 1902 nM T82739 C8FZ2L 118721003 Ki = 45 nM T82739 C0M4IQ 118721004 Ki = 20 nM T82739 CLRB29 118721005 Ki = 8 nM T82739 C9B1FX 118721007 Ki = 50 nM T82739 CRV5Y1 118721008 Ki = 5 nM T82739 CH6AQ9 118721009 Ki = 2 nM T82739 CHQ5P7 118987013 Ki = 42 nM T82739 C2V6PQ 122550396 IC50 = 8.5 nM T82739 C8NR0Y 122550417 IC50 = 0.7 nM T82739 C3W6DG 122551266 IC50 = 1.7 nM T82739 C5Y8IS 127025168 Ki = 7.5 nM T82739 CY03UC 127027302 Ki = 804 nM T82739 C18GDE 127027303 Ki = 317 nM T82739 CK0W2P 127027635 Ki = 59 nM T82739 CWJ0Y6 127027636 Ki = 55 nM T82739 C36DML 127029802 Ki = 150 nM T82739 CLJ40K 127029803 Ki = 120 nM T82739 CPC0M8 127031390 Ki = 550 nM T82739 C1BWV2 127035672 Ki = 22 nM T82739 CTMR64 127035685 Ki = 64 nM T82739 CVRY56 127036086 Ki = 8 nM T82739 C9B6LT 127037264 Ki = 9.93 nM T82739 C60HLK 127037469 Ki = 136 nM T82739 C85ROH 127041472 IC50 > 100000 nM T82739 CSB70O 129103433 IC50 = 4 nM T82739 C1QNA4 129103439 IC50 = 19 nM T82739 C82CEQ 129103576 IC50 = 900 nM T82739 CWXN62 129103630 IC50 = 9 nM T82739 CE2NT3 134130030 IC50 > 3000000 nM T82739 CT2RV6 134130781 IC50 = 2.4 nM T82739 CO13UB 134131040 IC50 = 1570 nM T82739 CWV3G6 134131077 IC50 = 153 nM T82739 CS8FV1 134131084 IC50 = 42.3 nM T82739 C1L3XV 134131107 IC50 = 8310 nM T82739 C92RTL 134131303 IC50 = 4.8 nM T82739 CSV13U 134131383 IC50 = 1210 nM T82739 CQOA40 134131498 IC50 = 53200 nM T82739 CL37SG 134131589 IC50 = 2 nM T82739 C6HTD5 135393470 IC50 = 11300 nM T82739 C7NA6E 135393474 IC50 > 50000 nM T82739 C4M5BF 135450980 Ki = 1300 nM T82739 CX62AU 135453491 Ki = 12 nM T82739 CYJ02B 135530536 Ki = 13 nM T82739 C8XC5J 135530568 Ki = 6 nM T82739 CBA90J 135532848 Ki = 4 nM T82739 CR6B1G 135532849 Ki = 6 nM T82739 CZHK63 135532851 Ki = 3 nM T82739 COA5Z0 135532896 Ki = 0.5 nM T82739 CW6DR2 135543006 Ki = 10 nM T82739 CTM4S0 135559104 Ki = 8 nM T82739 C3N1HW 135559111 Ki = 3 nM T82739 CYD5H1 135559116 Ki = 6 nM T82739 CD8XW3 135559124 Ki = 18 nM T82739 CZQ79E 135559125 Ki = 37 nM T82739 C90YUE 135559128 Ki = 65 nM T82739 C5DQ1E 135559129 Ki = 27 nM T82739 C4CMO6 136003658 Ki = 36 nM T82739 CM1LF3 136094796 Ki = 5 nM T82739 C1GPL0 136402490 Ki = 4820 nM T82739 CDQ62V 137637214 Ki = 3 nM T82739 C2K8JV 137639385 Ki = 0.25 nM T82739 C7EJ6B 137642984 Ki = 1.3 nM T82739 CG67RS 137643031 Ki = 0.06 nM T82739 CODW67 137644829 Ki = 45100 nM T82739 C83GDO 137646822 Ki = 0.44 nM T82739 C5SQZ6 137649699 Ki = 2.3 nM T82739 CCMQ19 137651042 Ki = 0.07 nM T82739 CN4ZT0 137651057 Ki = 0.39 nM T82739 C4M6NX 137651852 Ki = 0.21 nM T82739 CNX46H 137654508 Ki = 0.36 nM T82739 CMK09U 137655401 Ki = 0.15 nM T82739 CLQ5X7 137657674 Ki = 2.1 nM T82739 C8R7WM 137661862 Ki = 0.14 nM T82739 CUZ35A 138115400 IC50 = 6309.57 nM T82739 CO51HN 139030452 IC50 > 50000 nM T82739 CV86MX 145962597 IC50 = 1 nM T82739 C51YBM 145963085 IC50 = 1900 nM T82739 CE6C0A 145970642 Ki = 192 nM T82739 CZ1R3B 145982984 Ki = 0.02 nM T82739 C4HLX8 146029523 IC50 = 16700 nM T82739 CH59QO 155510375 Ki = 43190 nM T82739 CICU31 155511394 Ki = 277 nM T82739 CZR36C 155511554 IC50 = 79.43 nM T82739 CA81QV 155512709 Ki = 6380 nM T82739 C2VX3G 155512946 Ki = 6.3 nM T82739 C2CI8S 155513907 Ki = 2205 nM T82739 CYT20V 155514020 Ki > 50000 nM T82739 CAT98N 155514640 Ki > 10000 nM T82739 CG9H4N 155515624 Ki = 9090 nM T82739 C7ZM4R 155515728 Ki = 7405 nM T82739 CFRS54 155516565 Ki = 10390 nM T82739 C1ZSV0 155517054 Ki = 12550 nM T82739 CF96DM 155518671 Ki > 10000 nM T82739 C6NX4K 155519661 IC50 = 10 nM T82739 C4MS1B 155519676 IC50 = 794.33 nM T82739 C7DUX3 155520916 Ki > 10000 nM T82739 CH0N9A 155523885 Ki = 319 nM T82739 CYL8M0 155526377 Ki = 4640 nM T82739 CX7CO2 155527010 Ki = 600 nM T82739 CN3BH5 155527998 IC50 = 79.43 nM T82739 CHYW65 155528639 IC50 = 199.53 nM T82739 CI1FR2 155529536 Ki = 0.6 nM T82739 CD7O2G 155530095 IC50 = 794.33 nM T82739 C46AZL 155530642 Ki > 25000 nM T82739 C35QWO 155531023 IC50 = 398.11 nM T82739 CP8K2J 155531811 Ki = 10470 nM T82739 C0UR8Q 155531991 Ki = 12000 nM T82739 CIHM01 155535907 Ki > 100000 nM T82739 C12HON 155536142 IC50 = 199.53 nM T82739 C7JMK4 155538439 Ki = 800 nM T82739 C9QE5N 155538514 Ki = 3865 nM T82739 CRT3D4 155540148 Ki = 7245 nM T82739 CL90DN 155540666 Ki > 10000 nM T82739 CY6DK3 155540964 IC50 = 5.012 nM T82739 C4CHR9 155542229 Ki = 7920 nM T82739 C4P2GV 155543617 Ki > 25000 nM T82739 CU52QS 155545897 Ki > 10000 nM T82739 CH2S6R 155546346 Ki > 10000 nM T82739 C5MB9R 155547962 IC50 = 50.12 nM T82739 CLFB25 155548371 IC50 = 794.33 nM T82739 CSI5J1 155548907 Ki = 7270 nM T82739 CU9FL4 155551858 Ki > 50000 nM T82739 COM52R 155551892 IC50 = 79.43 nM T82739 CA5VG2 155552651 Ki = 24500 nM T82739 C5S6HO 155553129 Ki = 6950 nM T82739 CJ3FI5 155553630 IC50 = 1258.93 nM T82739 C5TV4J 155554082 Ki = 8246 nM T82739 CU8LR3 155555208 Ki > 25000 nM T82739 CSW48V 155557718 IC50 = 19.95 nM T82739 CXL5D4 155558368 Ki = 48690 nM T82739 CNZ1K5 155559920 Ki > 10000 nM T82739 C3SXY1 155561904 Ki = 64397 nM T82739 CX5O7K 155562968 Ki = 540 nM T82739 CM8XB1 155565537 IC50 = 100 nM T82739 CP4F1U 155567613 Ki = 32000 nM T82739 CEZ8B9 155568406 Ki > 50000 nM T82739 CK0EA2 155568484 Ki = 701 nM T82739 CL2S7B 90655701 Ki = 320000 nM T82739 D02AVL 18376720 Ki = 45 nM T82739 D02PAU 16731825 Ki = 1000 nM T82739 D02YIW 1794 IC50 > 50000 nM T82739 D05ZIP 674656 IC50 = 6200 nM T82739 D07ZRG 46899577 Ki = 8.3 nM T82739 D08KCA 72429 IC50 = 40000 nM T82739 D08OCS 699665 IC50 = 6100 nM T82739 D08WQJ 700133 IC50 = 18800 nM T82739 D0A8WP 447732 Ki = 2500 nM T82739 D0IU5E 716930 IC50 = 12300 nM T82739 D0J5VK 67145 IC50 = 67900 nM T82739 D0JU9N 6914623 Ki > 2800 nM T82739 D0K7YL 447476 Ki = 1.9 nM T82739 D0M4VZ 10456438 IC50 = 31 nM T82739 D0ON2Z 204102 Ki > 2300 nM T82739 D0R9CH 3400921 Ki = 37 nM T82739 D0X1OY 674628 IC50 = 5700 nM T82739 D0Y5IQ 44255320 IC50 = 10000 nM T45593 D05YBZ 7083 Ki = 69 nM T45593 D05TPI 72276 IC50 >= 200000 nM T45593 D07SDQ 969516 IC50 = 3500 nM T45593 D0U2BH 65064 IC50 = 1800 nM T45593 C2KJI7 3883 Ki = 2.5 nM T45593 C0VAW3 13735 IC50 = 69 nM T45593 CYX3S5 65043 IC50 = 69 nM T45593 C39BCE 68275 IC50 < 3000 nM T45593 CO41FC 964143 Ki = 789.8 nM T45593 CJ0O1B 1588443 IC50 = 380 nM T45593 CO1ZV8 2306524 Ki = 522.1 nM T45593 CY28LS 5293755 Ki = 617.6 nM T45593 C5ZS3K 5713403 Ki = 528.5 nM T45593 CZ9Q1O 5928757 Ki = 362.5 nM T45593 CQ3S8L 6450842 Ki = 261.5 nM T45593 CFXW58 11631766 Ki = 1410 nM T45593 C7EBU1 11776207 IC50 > 10000 nM T45593 CLV24A 14214498 IC50 = 1400 nM T45593 C62KEJ 14837578 IC50 = 710 nM T45593 CN0Y8F 15504852 IC50 = 13 nM T45593 CN9U3G 16049314 IC50 = 246 nM T45593 CWUS28 22361008 IC50 > 10000 nM T45593 CCL0P8 24858429 IC50 = 1635 nM T45593 CYDL23 24952085 IC50 = 440 nM T45593 C1RB4M 24966387 IC50 = 1200 nM T45593 C0BN8L 42643531 IC50 = 4 nM T45593 CD80XQ 54581735 IC50 = 80 nM T45593 C4FZ5A 56950118 Ki = 13 nM T45593 C90MUF 57176479 Ki = 599 nM T45593 C2K6JT 57379031 EC50 = 24 nM T45593 CTA24H 57578199 IC50 = 1700 nM T45593 CC8ZH7 58660303 IC50 > 10000 nM T45593 CU1D5F 58795397 Ki = 797.8 nM T45593 CQU9W0 66556402 Ki = 191.3 nM T45593 CJ4R7E 66571561 IC50 = 660 nM T45593 CAJ6B8 67973277 EC50 = 325 nM T45593 C2ZCF9 67973354 EC50 = 169 nM T45593 C9JMF7 68551830 IC50 = 910 nM T45593 CXS67Z 68552247 IC50 = 580 nM T45593 CWE58F 68553100 IC50 = 690 nM T45593 CH54DU 68553676 IC50 = 600 nM T45593 CY8HE3 68553756 IC50 = 420 nM T45593 C1LYJ4 68553873 IC50 > 10000 nM T45593 CAG5N8 68554590 IC50 = 2000 nM T45593 CSQ53N 68555084 IC50 = 520 nM T45593 CEI5O1 68555350 IC50 = 320 nM T45593 CNCS47 68556083 IC50 = 1400 nM T45593 CN2QL6 68556085 IC50 = 920 nM T45593 CR4VM9 70686684 Ki = 1428 nM T45593 CD1PU4 70688786 Ki = 17 nM T45593 C59PES 70694381 Ki = 0.48 nM T45593 CZ3QF7 70697093 Ki = 112 nM T45593 CW0ZX3 71452100 IC50 = 2 nM T45593 CUP70I 71453931 IC50 = 1251 nM T45593 C7EX1K 71457447 IC50 = 17 nM T45593 CM5E3R 71457448 IC50 = 2 nM T45593 C3GPE7 71457449 IC50 = 4707 nM T45593 C7XML1 71457851 IC50 = 5.1 nM T45593 C4AK0O 71459256 IC50 = 42 nM T45593 CQ0FG2 71459258 IC50 = 7469 nM T45593 CYN3M8 71461086 IC50 = 1591 nM T45593 CW1E7U 71462763 IC50 = 6 nM T45593 CM6R2W 71463212 IC50 = 1.41 nM T45593 CLVB69 73294880 IC50 = 13 nM T45593 CGZK85 73296378 IC50 = 2 nM T45593 C9L3VR 73296809 IC50 = 2 nM T45593 C2S9PZ 73296810 IC50 = 5 nM T45593 C4XR1C 73297137 IC50 = 1 nM T45593 CCPI94 73297139 IC50 = 3 nM T45593 CE9X5J 86713212 IC50 = 420 nM T45593 C45CME 89681657 IC50 > 10000 nM T45593 C3R4PD 89970609 IC50 = 330 nM T45593 C06FNJ 89970660 IC50 = 610 nM T45593 CE1IW4 89970765 IC50 = 700 nM T45593 CEF8J5 90040128 IC50 = 5 nM T45593 CD48HU 90277509 IC50 > 10000 nM T45593 CX28SL 90644922 IC50 = 2 nM T45593 CHD0Z7 90644923 IC50 = 79 nM T45593 CYPJ75 90644924 IC50 = 8 nM T45593 CTL20G 102196384 IC50 > 10000 nM T45593 C5PBW3 102398558 IC50 > 10000 nM T45593 C5W7PM 118713185 IC50 > 10000 nM T45593 CQ07AH 118713186 IC50 > 10000 nM T45593 C5OFH2 118713187 IC50 > 10000 nM T45593 C9ZGB4 118713188 IC50 > 10000 nM T45593 C7Z2GA 118713189 IC50 > 10000 nM T45593 C03URO 118713190 IC50 > 10000 nM T45593 CYK30H 118713191 IC50 > 10000 nM T45593 CK53ME 118713192 IC50 > 10000 nM T45593 C35IDH 118713193 IC50 < 290 nM T45593 CM7UC8 118713194 IC50 > 10000 nM T45593 C5C8LX 118713195 IC50 = 300 nM T45593 C1RH3Y 118713196 IC50 = 1600 nM T45593 CB03DR 122182244 Ki = 212.4 nM T45593 CI6WT0 122182245 Ki = 431.7 nM T45593 C3X5KJ 122182246 Ki = 364 nM T45593 CT5G1Q 122182247 Ki = 1116.2 nM T45593 CCT7H6 122182248 Ki = 858.8 nM T45593 CML3T5 122182249 Ki = 853.5 nM T45593 CMO1C3 122182250 Ki = 169 nM T45593 CIT52U 122182251 Ki = 53.7 nM T45593 C19GJH 122182252 Ki = 35.1 nM T45593 CUOB01 122182253 Ki = 48 nM T45593 CW2V5B 122182254 Ki = 682.4 nM T45593 C75OCP 122182255 Ki = 717.6 nM T45593 CVH2T0 122182256 Ki = 229.1 nM T45593 CKQF12 122182257 Ki = 374 nM T45593 C7AUF8 122182258 Ki = 239.7 nM T45593 C7BXY4 122182259 Ki = 90 nM T45593 CCEL74 122182260 Ki = 188 nM T45593 C32GEV 122182261 Ki = 263.2 nM T45593 CWIT38 122182262 Ki = 257 nM T45593 CMVS36 122182263 Ki = 204.3 nM T45593 CLW95X 122182264 Ki = 131.1 nM T45593 C4TNB1 122182265 Ki = 465.1 nM T45593 CQ4R0K 122182266 Ki = 38.3 nM T45593 C5C8FY 122182267 Ki = 1756.7 nM T45593 C7NV9G 122182268 Ki = 27.1 nM T45593 CU3NJ6 122182269 Ki = 208.7 nM T45593 CS84HC 122182270 Ki = 121.5 nM T45593 C8EYO3 122182271 Ki = 590.5 nM T45593 CFV32E 122182272 Ki = 72.4 nM T45593 C1LHQ2 122182273 Ki = 318.1 nM T45593 C24PHB 122182274 Ki = 228.6 nM T45593 C1U3FZ 122182275 Ki = 354.6 nM T45593 CX5NB4 122182276 Ki = 151.7 nM T45593 CAU9H6 122182277 Ki = 630.3 nM T45593 C2RB1F 122182278 Ki = 80.1 nM T45593 CTMV35 122182279 Ki = 455.7 nM T45593 CO54NG 134133007 IC50 = 230 nM T45593 C4G8CN 136259624 IC50 = 970 nM T45593 C0PX2K 145968691 IC50 = 12900 nM T45593 C4R3UA 145978145 IC50 = 27200 nM T45593 CYB0T8 155552280 Ki = 120 nM T45593 D05CCT 4139 EC50 = 130 nM T45593 D0O5FK 10171487 IC50 = 3255 nM T45593 D0T3PW 5281672 IC50 = 1200 nM T45593 D0Z7EL 5280647 IC50 < 3000 nM T62292 D07JVL 3016 Ki = 17 nM T62292 D0L9GG 2118 EC50 = 69 nM T62292 D0T1WN 5732 Ki = 400 nM T62292 D0CH7C 57336276 Ki = 489 nM T62292 D0HO2T 23581869 Ki = 1.3 nM T62292 D0Z9HW 23630026 Ki = 3.1 nM T62292 C4PAD5 5255267 Ki = 858 nM T62292 C1Z6YU 9821389 Ki = 12 nM T62292 CCX58U 9865233 Ki = 1.8 nM T62292 C7BA0Z 9908880 Ki = 0.7 nM T62292 C1VRB9 9951530 EC50 = 23 nM T62292 CPC3U1 9971547 Ki > 300 nM T62292 CUT5W8 9976743 EC50 = 33 nM T62292 CUSM85 10221761 Ki = 0.5 nM T62292 C15NXT 10926766 EC50 = 3826 nM T62292 CK1S7J 10927005 EC50 = 367 nM T62292 CWK02D 10936672 EC50 = 424 nM T62292 C09PCZ 10971225 EC50 = 500 nM T62292 C74SOK 11001453 EC50 = 935 nM T62292 CJB1V2 11035207 EC50 = 394 nM T62292 CBV36I 11047145 EC50 = 213 nM T62292 C8B7TF 11067772 EC50 = 116 nM T62292 CAU9O6 11142977 EC50 = 117 nM T62292 CWO70Q 11673720 Ki = 14 nM T62292 CX7G9K 11759134 EC50 = 344 nM T62292 CL4XD0 11783674 EC50 = 20 nM T62292 CYD2G3 11809547 EC50 = 71 nM T62292 C1ZXE0 15951053 Ki = 8545 nM T62292 C6HY4N 21065276 Ki = 272 nM T62292 C5R3SB 21930923 Ki = 96 nM T62292 CPM7G9 25093403 Ki = 2666 nM T62292 C8E3KW 25093404 Ki = 1864 nM T62292 CZK75V 44364548 EC50 = 425 nM T62292 C0FN6W 44364725 EC50 = 375 nM T62292 CE8F3Y 44364734 EC50 = 265 nM T62292 COH5G6 44364735 EC50 = 119 nM T62292 C2VHW7 44364747 EC50 = 148 nM T62292 CZL2P0 44364907 EC50 = 65 nM T62292 CCX08E 44364918 EC50 = 242 nM T62292 C6AO8S 44561476 Ki = 255 nM T62292 CLQZ42 44561477 Ki = 198 nM T62292 C27YZH 88286432 Ki = 1000 nM T62292 CQ91VU 118278442 Ki = 24 nM T62292 CH0D4J 130439777 Ki = 660 nM T62292 C56XBU 130439778 Ki = 63000 nM T62292 C9N8LW 130439889 Ki = 480 nM T62292 D06SOQ 6918451 Ki = 0.61 nM T62292 D09IHE 6918583 Ki = 0.77 nM T62292 D0D9RF 9927764 Ki = 18.7 nM T62292 D0E7PY 11624499 Ki = 80 nM T62292 D0GQ2G 5311418 Ki = 25.8 nM T62292 D0O9MG 5311203 Ki = 17 nM T21782 D06RGG 5819 IC50 > 50000 nM T21782 D0S6JG 5920 IC50 = 3600 nM T21782 D0J6XC 5803 IC50 = 25000 nM T21782 D0WM6E 160565 IC50 = 32000 nM T21782 CLSK17 5804 IC50 = 17000 nM T21782 CPR38J 92859 IC50 = 6300 nM T21782 C2VED9 107564 IC50 > 50000 nM T21782 CHM8L9 71185084 IC50 = 1200 nM T21782 CTN04E 71185155 IC50 = 9700 nM T21782 CU8KD9 71185156 IC50 = 1200 nM T21782 CB49TE 71185169 IC50 = 1000 nM T21782 CDLU47 71185374 IC50 = 1500 nM T21782 CB8R1S 71185474 IC50 = 6000 nM T21782 CP6Z7Y 71185477 IC50 = 1400 nM T21782 CNU60F 71185540 IC50 = 1000 nM T21782 CNR1C2 71487227 IC50 = 1900 nM T21782 CPM3Q9 71487297 IC50 = 2700 nM T21782 CD1T9B 71487299 IC50 = 2900 nM T21782 C2YMT4 71487301 IC50 = 3100 nM T21782 C06COQ 71487363 IC50 = 3700 nM T21782 CQV8L7 71487428 IC50 = 11000 nM T21782 CTB4V0 71583751 IC50 > 50000 nM T21782 C6UV0P 71583752 IC50 > 50000 nM T21782 C6E7DR 71583865 IC50 > 50000 nM T21782 C2CD7N 71583866 IC50 > 50000 nM T21782 CA2TH8 71583867 IC50 = 14000 nM T21782 CGX57L 71583868 IC50 = 8600 nM T21782 C76GXY 71583869 IC50 = 6500 nM T21782 CPI36K 71583870 IC50 = 2900 nM T21782 CH3J9Z 71583871 IC50 = 6000 nM T21782 CM4LY2 71583975 IC50 = 1300 nM T76369 D0E6YQ 1935 IC50 > 100000 nM T76369 D0NS6H 3152 IC50 > 100000 nM T76369 D0Y3KG 3121 Ki = 363000 nM T76369 D0B6IZ 137905 Ki = 2.1 nM T76369 D0W0VD 3885 Ki = 1220 nM T76369 D02UOE 160142 Ki = 2530 nM T76369 C13GAP 255 IC50 = 140 nM T76369 CXU4W0 650 Ki > 100000 nM T76369 C0RFA2 3102 Ki > 100000 nM T76369 C4IU5T 6889 Ki = 31700 nM T76369 C6B1HI 9905 IC50 = 4 nM T76369 C25CYL 10434 Ki > 100000 nM T76369 C47FYB 10662 Ki > 100000 nM T76369 CZP3G7 11100 Ki > 100000 nM T76369 COGY52 11321 Ki = 36000 nM T76369 C7U0TW 11747 Ki > 100000 nM T76369 C53FYO 11840 Ki > 100000 nM T76369 CKR3L9 12116 Ki > 100000 nM T76369 CU5KZ0 13005 Ki > 100000 nM T76369 CJ2GH1 13006 Ki > 100000 nM T76369 CG1LI5 14313 Ki > 100000 nM T76369 C4FW7E 18475 Ki > 100000 nM T76369 C7S3JO 26257 Ki = 3 nM T76369 C38JQX 31261 Ki > 100000 nM T76369 CN8A2G 38296 Ki > 100000 nM T76369 C7HE8W 38333 Ki > 100000 nM T76369 C0VK3I 39834 Ki > 100000 nM T76369 C8Z6TM 43402 Ki > 100000 nM T76369 CUNJ73 61209 Ki > 100000 nM T76369 C6U7FB 62539 Ki > 100000 nM T76369 CEKW96 68115 Ki = 125.89 nM T76369 CL5B7Z 68119 Ki = 1170 nM T76369 C27NHT 69147 Ki > 100000 nM T76369 CN0ID1 69282 Ki > 100000 nM T76369 CW54JA 69288 Ki > 100000 nM T76369 C6BEN0 70945 Ki > 100000 nM T76369 CV8R4B 76561 Ki > 100000 nM T76369 CVJ78Y 79690 Ki = 46.6 nM T76369 CAPG58 87502 Ki = 77.6 nM T76369 C0EH3Z 88695 Ki = 26900 nM T76369 C70KGR 92036 Ki = 3300 nM T76369 C13IQL 93772 Ki > 100000 nM T76369 C7JEN0 94320 IC50 = 49860 nM T76369 C8YU9Z 95415 Ki > 100000 nM T76369 CH91PI 95447 Ki > 100000 nM T76369 CO0QF3 97313 Ki = 942 nM T76369 C6L8SK 102135 IC50 = 22360 nM T76369 CR3E9L 103786 Ki > 100000 nM T76369 CFG6D1 111253 IC50 > 100000 nM T76369 C7KJ3B 114917 Ki = 26250 nM T76369 C20LIY 136371 Ki > 100000 nM T76369 CTU83D 137777 Ki = 22800 nM T76369 CHAN02 138508 Ki = 8060 nM T76369 CYX5V0 142278 Ki > 100000 nM T76369 C5X1YU 160254 Ki = 544 nM T76369 CXG41E 163959 Ki = 355000 nM T76369 C4IRY2 164676 Ki = 6890 nM T76369 CB9GM4 176443 IC50 = 2 nM T76369 CD35GB 181715 Ki = 707000 nM T76369 C6W8MB 219592 Ki > 100000 nM T76369 COQ09W 219605 Ki = 1550 nM T76369 C25BHS 222475 Ki > 100000 nM T76369 CN35KE 222570 Ki > 100000 nM T76369 C93DSW 222958 IC50 = 10 nM T76369 CP4W3S 229680 Ki = 3080 nM T76369 C2SQH9 232004 Ki > 100000 nM T76369 C0KV5M 236566 Ki > 100000 nM T76369 CE6U1D 237515 Ki = 4.8 nM T76369 C92OSL 241331 Ki = 53900 nM T76369 C1IW3D 261836 Ki > 100000 nM T76369 CHP1J7 262695 Ki > 100000 nM T76369 CDL3E1 262696 Ki > 100000 nM T76369 CPL6E4 272516 Ki = 32.1 nM T76369 CBV0N9 275005 Ki = 212 nM T76369 C18XWV 291540 Ki > 100000 nM T76369 CH52BM 306215 Ki > 100000 nM T76369 CKS3U9 366710 Ki = 34100 nM T76369 CKP61X 368568 Ki = 1054 nM T76369 CTWM69 586418 Ki > 100000 nM T76369 CH1E7N 590628 Ki > 100000 nM T76369 C4TE6S 597830 Ki > 100000 nM T76369 CCJQ96 599378 Ki = 170 nM T76369 COW64L 988563 Ki = 13700 nM T76369 C79KSZ 1009717 Ki > 100000 nM T76369 CAP82W 1103353 Ki > 100000 nM T76369 CB8I0Q 1133380 Ki > 100000 nM T76369 C21KSG 1137588 Ki > 100000 nM T76369 CF46TV 1167776 Ki > 100000 nM T76369 CN8BI5 1222869 Ki > 100000 nM T76369 CWTV42 1713189 Ki = 4350 nM T76369 C0EX9G 1755771 Ki = 66 nM T76369 CB0ZP3 1812008 Ki = 9800 nM T76369 C3FQD8 1906162 Ki > 100000 nM T76369 C3O6MN 1972026 Ki > 100000 nM T76369 CF37ZA 2147394 Ki = 610 nM T76369 CJD8B3 2305233 Ki = 2650 nM T76369 C0OZQ2 2731126 Ki > 100000 nM T76369 CNKV06 2731127 Ki = 1620 nM T76369 CEM2C8 2731732 Ki = 19500 nM T76369 C2HOC5 2731733 Ki = 1880 nM T76369 CVC36I 2731902 Ki = 1420 nM T76369 CG62CN 2731904 Ki = 36000 nM T76369 CVD82J 2734800 Ki = 1660 nM T76369 C9R5LQ 2749125 Ki = 2630 nM T76369 C84DSN 2749126 Ki = 107 nM T76369 C84VWR 2784639 Ki = 5380 nM T76369 CDCB42 2786143 Ki = 1540 nM T76369 C43YAR 2835143 Ki > 100000 nM T76369 C1AM0S 3114312 Ki = 1560 nM T76369 C61RSW 3126152 Ki > 100000 nM T76369 CCP07Y 3264931 Ki > 100000 nM T76369 CB21VL 3321360 Ki > 100000 nM T76369 CZV6G2 3329233 Ki > 100000 nM T76369 C6NH9P 3469206 Ki > 100000 nM T76369 C10GCK 3527426 Ki = 1690 nM T76369 C3T1CV 3531512 Ki > 100000 nM T76369 C5UM2D 3821945 Ki = 8 nM T76369 CU17BR 4088910 Ki > 100000 nM T76369 C8CFN7 4118889 Ki > 100000 nM T76369 CC1GF9 4338240 Ki = 580 nM T76369 C8KV7I 4350924 Ki > 100000 nM T76369 C0V6QI 4369935 Ki > 100000 nM T76369 C0GS5T 4381638 Ki > 100000 nM T76369 C42FGN 4384851 Ki = 7.5 nM T76369 CQ46SJ 4427802 Ki > 100000 nM T76369 CN9C3V 4513067 Ki = 55300 nM T76369 C5NJ3A 5004413 Ki > 100000 nM T76369 CNMY06 5038499 Ki > 100000 nM T76369 CWCG89 5080545 Ki > 100000 nM T76369 CK5XC9 5235003 Ki > 100000 nM T76369 CMJ30V 5353845 IC50 = 5000 nM T76369 CY6D5H 9821458 IC50 = 1000 nM T76369 CZ10UR 9905153 IC50 = 2000 nM T76369 CHT5U3 10044204 IC50 = 6000 nM T76369 CTZ42X 10337211 IC50 = 3470 nM T76369 CWE41Q 10655805 Ki = 6.65 nM T76369 CE64FC 10661387 Ki = 17.7 nM T76369 CF28NJ 10879668 Ki = 7.6 nM T76369 CH49NV 10899196 Ki = 102 nM T76369 CP93JE 10902085 Ki = 0.84 nM T76369 C7NZY9 11009341 Ki = 21000 nM T76369 C1P3HT 11226329 Ki > 100000 nM T76369 CC3D2X 11245953 Ki = 2.2 nM T76369 CYJ2M4 11278743 IC50 = 300 nM T76369 CSD58O 11280423 Ki = 7 nM T76369 C8GX1Y 11322015 Ki = 363.08 nM T76369 CI68UO 11393923 IC50 = 1000 nM T76369 C1JAC5 11425923 Ki = 398 nM T76369 CU94ZT 11484453 IC50 = 140 nM T76369 CG2B7X 11631387 IC50 = 30 nM T76369 C0QJ9O 11652690 IC50 = 30 nM T76369 C57KVO 11674428 IC50 = 10 nM T76369 CG7O5E 11695972 IC50 = 200 nM T76369 CV74JA 11696246 IC50 = 500 nM T76369 CAG6H2 11709766 IC50 = 250 nM T76369 CY58GA 11739291 IC50 = 200 nM T76369 CCQN45 11805526 Ki = 26 nM T76369 CMV1U9 11991810 IC50 = 7000 nM T76369 CVK4C5 11991896 IC50 = 200 nM T76369 CI9R2Y 11991988 IC50 = 100 nM T76369 CV2M3J 12057101 Ki = 0.302 nM T76369 CKG7A0 12222796 Ki > 100000 nM T76369 CJ65IL 12305517 IC50 = 10530 nM T76369 C8B5LO 13780062 Ki = 2.19 nM T76369 C3YOX2 13827082 Ki > 100000 nM T76369 C4CR1L 13827083 Ki > 100000 nM T76369 CH27JR 14609844 Ki = 0.328 nM T76369 CKX0P8 14610645 Ki = 1223 nM T76369 CA0E1T 14610646 Ki = 25.1 nM T76369 CI68WP 14707309 IC50 = 23610 nM T76369 CSI6M2 14828209 Ki = 131 nM T76369 CBA8U6 14856680 Ki = 23.8 nM T76369 CJ6H8G 14856681 Ki = 18.9 nM T76369 CL2C7Y 15044210 Ki = 870 nM T76369 C3UXC5 16084218 IC50 = 1960 nM T76369 C45MVX 16110641 IC50 > 100000 nM T76369 CC9N1G 16110651 IC50 = 500 nM T76369 CO94HF 16110652 IC50 = 400 nM T76369 CLC13N 16110653 IC50 = 200 nM T76369 COK20Z 16110654 IC50 = 600 nM T76369 C0H5RW 16110655 IC50 = 900 nM T76369 CS0VQ6 16110656 IC50 = 6000 nM T76369 COL87N 16110658 IC50 = 3000 nM T76369 C0KT5Q 16110666 IC50 = 30000 nM T76369 CVC17D 16110699 IC50 > 100000 nM T76369 C7O1KM 16110701 IC50 = 200 nM T76369 C97PDA 16110708 IC50 = 2000 nM T76369 C8P1JE 16110710 IC50 = 2000 nM T76369 CX3LI0 16110711 IC50 = 34000 nM T76369 C42XSZ 16110715 IC50 > 100000 nM T76369 CBH6F1 16110717 IC50 > 100000 nM T76369 CWV39U 16110722 IC50 = 8000 nM T76369 C5W1CT 16110723 IC50 = 30000 nM T76369 CPG32I 16307342 Ki > 100000 nM T76369 CXQO59 16324698 Ki > 100000 nM T76369 CX5UT9 16735161 IC50 = 200 nM T76369 C3KF9Y 16736226 IC50 = 2000 nM T76369 CR76ET 16737951 IC50 = 1200 nM T76369 C8G9AL 16756850 IC50 > 10000 nM T76369 CKX36J 17479504 Ki > 100000 nM T76369 CBG35K 17485200 Ki > 100000 nM T76369 C2OF8S 18471933 Ki > 100000 nM T76369 CG5DA4 22109309 Ki > 100000 nM T76369 C1IQ9L 22486206 IC50 = 5 nM T76369 CM3Y1I 22574246 Ki > 100000 nM T76369 CET65Y 22772978 Ki > 100000 nM T76369 C3F1EG 22772980 Ki > 100000 nM T76369 CKUJ63 22772981 Ki > 100000 nM T76369 C6WY3U 23669322 Ki > 100000 nM T76369 CX1G5Y 24319385 Ki > 100000 nM T76369 C0LP8T 24445964 Ki > 100000 nM T76369 CNF01W 24748349 IC50 = 70 nM T76369 CF9E1W 24748380 IC50 = 3000 nM T76369 COE7A6 24799115 IC50 > 100000 nM T76369 C3A6LN 24799306 IC50 = 7000 nM T76369 CMEC63 24799824 IC50 = 16 nM T76369 C59EGV 24799998 IC50 > 100000 nM T76369 C5V6OE 24800169 IC50 = 270 nM T76369 CU9Y3V 24800335 IC50 = 100 nM T76369 C5MK9H 24800509 IC50 = 17000 nM T76369 CSB1L8 24800681 IC50 > 100000 nM T76369 CLC63B 24800683 IC50 = 90000 nM T76369 CI67RX 24800861 IC50 = 2400 nM T76369 CT5C9E 24801041 IC50 = 37000 nM T76369 C0RT3I 24801044 IC50 = 26000 nM T76369 C8WGD9 24801560 IC50 = 26 nM T76369 CQNB75 24825630 Ki > 100000 nM T76369 C2EPR4 24948911 IC50 > 100000 nM T76369 C0MC4D 24948914 IC50 = 120 nM T76369 CSA71C 24949075 IC50 = 2000 nM T76369 CGK9I3 24949076 IC50 = 200 nM T76369 C79BEQ 24949227 IC50 = 12000 nM T76369 CGO7P4 24950363 IC50 > 100000 nM T76369 CS8H1V 24950364 IC50 = 8000 nM T76369 C90WNP 24950523 IC50 = 30000 nM T76369 C5O4JY 24950525 IC50 = 800 nM T76369 CO37IU 24950526 IC50 = 11000 nM T76369 CUH23T 24950528 IC50 > 100000 nM T76369 CY2NW6 24950843 IC50 = 40 nM T76369 C9BYQ6 24950844 IC50 = 40000 nM T76369 CLW02V 24951001 IC50 = 30 nM T76369 C4MXB8 24951004 IC50 = 150 nM T76369 CIF25O 24951005 IC50 = 40000 nM T76369 CFJW54 24951156 IC50 = 400 nM T76369 CDJ4N0 24951159 IC50 = 3000 nM T76369 C7O2MR 24951162 IC50 = 40000 nM T76369 C3GC9N 24951316 IC50 = 1500 nM T76369 C7NZ2X 24951318 IC50 > 100000 nM T76369 CUDP87 24951320 IC50 > 100000 nM T76369 CWID81 25325634 Ki > 100000 nM T76369 C8HQZ7 44157144 Ki > 100000 nM T76369 C4HL5B 44157145 Ki > 100000 nM T76369 CPM08L 44157218 Ki > 100000 nM T76369 CD5XW6 44157219 Ki > 100000 nM T76369 CU8EQ7 44157220 Ki > 100000 nM T76369 C2PZN0 44157221 Ki > 100000 nM T76369 CSW49B 44157293 Ki > 100000 nM T76369 CO30PI 44157294 Ki > 100000 nM T76369 C47BWL 44157295 Ki > 100000 nM T76369 CA80TE 44157296 Ki > 100000 nM T76369 CGZW85 44157297 Ki > 100000 nM T76369 C7GK9S 44157298 Ki > 100000 nM T76369 CUA79M 44157370 Ki > 100000 nM T76369 C8NK1F 44157371 Ki > 100000 nM T76369 CJXT82 44157372 Ki > 100000 nM T76369 C4UWK6 44157373 Ki > 100000 nM T76369 CZY1Q3 44157374 Ki > 100000 nM T76369 CWIH19 44157375 Ki > 100000 nM T76369 CLS06F 44157439 Ki > 100000 nM T76369 C4R5HG 44157440 Ki > 100000 nM T76369 C03DWN 44157441 Ki > 100000 nM T76369 C3U2AW 44157442 Ki > 100000 nM T76369 CR6DQ1 44157443 Ki > 100000 nM T76369 CKD82Y 44157512 Ki > 100000 nM T76369 CH4T2Z 44157513 Ki > 100000 nM T76369 C8RTA7 44389776 IC50 = 5 nM T76369 CS1JH5 44389963 IC50 = 20000 nM T76369 C84ISX 44389973 IC50 = 20000 nM T76369 CJ91NL 44391726 IC50 = 80 nM T76369 C0C2DX 44428836 Ki > 100000 nM T76369 CZS9U1 44428842 Ki > 100000 nM T76369 CWR3Y1 44428843 Ki > 100000 nM T76369 CUT0H7 44428844 Ki > 100000 nM T76369 C10PFH 44554611 IC50 = 10000 nM T76369 CL6C1X 44554613 IC50 = 700 nM T76369 C6KCQ1 44554787 IC50 = 60 nM T76369 C7M5YB 44569835 Ki = 0.3981 nM T76369 CS61ZR 44569836 Ki = 0.3981 nM T76369 CT3U4M 44569837 Ki = 0.5012 nM T76369 C6IEG1 44569871 Ki = 0.6026 nM T76369 C95PNJ 44569872 Ki = 0.6026 nM T76369 CZF6X0 44569873 Ki = 3.311 nM T76369 C6TQF9 44569874 Ki = 0.7079 nM T76369 C7KS9O 44569875 Ki = 1 nM T76369 C5KO9F 44569911 Ki = 6.457 nM T76369 CB78NA 44569912 Ki = 6.026 nM T76369 CXUP02 44583034 Ki > 100000 nM T76369 CEK3P8 44583159 Ki > 100000 nM T76369 C7IJ3C 49857726 Ki = 279 nM T76369 C04NYX 49857906 Ki > 100000 nM T76369 CDT4Y6 49857907 Ki = 437 nM T76369 C5XS3G 49857908 Ki = 1034 nM T76369 CHRB62 49857909 Ki = 1244 nM T76369 CV7J6X 49857910 Ki > 100000 nM T76369 CYU39N 49857911 Ki > 100000 nM T76369 C5WZL0 49857912 Ki = 756 nM T76369 CCG80U 49858100 Ki > 100000 nM T76369 CCN05H 49858101 Ki = 381 nM T76369 C6S0TB 52944501 IC50 = 26260 nM T76369 CY67HJ 52948155 IC50 = 10970 nM T76369 C5FE4Z 52948907 IC50 = 34 nM T76369 C4OF7Q 53483972 IC50 > 100000 nM T76369 C1QWH9 56931986 IC50 > 100000 nM T76369 CO29WI 71508729 Ki = 17.8 nM T76369 CM93WB 92131904 Ki = 468000 nM T76369 CS1GL7 96359892 Ki = 24800 nM T76369 CDBZ20 102189779 Ki = 0.417 nM T76369 C2CL6P 127030256 IC50 > 100000 nM T76369 CV6B4Z 127030257 IC50 = 12310 nM T76369 CZ0NI1 127030258 IC50 = 25090 nM T76369 C3DL4M 127031478 IC50 = 9130 nM T76369 C2YD1M 127031479 IC50 = 6990 nM T76369 CF0OI3 127034386 IC50 = 20410 nM T76369 C1ZP4G 130431469 IC50 > 10000 nM T76369 CMA35H 130431481 IC50 > 10000 nM T76369 CX59ME 133561407 Ki = 2.4 nM T76369 C8R0BI 137633433 Ki = 148 nM T76369 CFP68C 137635195 Ki = 45.3 nM T76369 CRO26U 137638968 Ki = 4.7 nM T76369 C56IMJ 137643802 Ki = 4.9 nM T76369 C0N3LP 137644595 Ki = 12.9 nM T76369 CBXV07 137652900 Ki = 16.1 nM T76369 CT9IF1 137657377 Ki = 15.6 nM T76369 C1UAZ3 137660095 Ki = 4.44 nM T76369 CEP6R2 137660441 Ki = 14.3 nM T76369 C7YDE3 145951659 IC50 > 100000 nM T76369 C0IS6K 145966157 Ki = 1871 nM T76369 C7HQ2O 145966235 Ki = 12.2 nM T76369 CH3W2Y 145966354 Ki = 102 nM T76369 C3TB2M 145966935 Ki = 25.9 nM T76369 CFT18Y 145969150 Ki = 2425 nM T76369 CQ9G1T 145972810 Ki = 31.9 nM T76369 C0V5WI 145974492 Ki = 48.7 nM T76369 CKD57H 145974917 Ki >= 10000 nM T76369 C6CQI9 145976186 Ki = 42.5 nM T76369 C60ICV 145976488 Ki = 4204 nM T76369 C6W2ZB 145976588 Ki = 14.4 nM T76369 CPL3T8 145977135 Ki = 42 nM T76369 C90CJY 145978164 Ki = 495 nM T76369 CVG8B2 145985484 Ki = 92.3 nM T76369 CQ61NL 145993296 Ki = 3.6 nM T76369 D00ANJ 1897797 Ki = 10 nM T76369 D00CKY 24951315 IC50 = 100 nM T76369 D00IAK 44455840 IC50 = 5.4 nM T76369 D00PLH 44428832 Ki = 230 nM T76369 D00ULT 10609180 IC50 = 10 nM T76369 D01HRG 12884 Ki = 23 nM T76369 D01HZN 44428835 Ki = 1000 nM T76369 D01NDE 11493344 Ki = 7.413 nM T76369 D01NWS 24801394 IC50 = 4.5 nM T76369 D01VAU 123493 Ki = 1540 nM T76369 D01VCS 44428837 Ki = 5650 nM T76369 D01XGP 123358 Ki = 5240 nM T76369 D02BDL 8433 Ki = 26000 nM T76369 D02ENI 10293363 IC50 = 10000 nM T76369 D02GJG 11043027 Ki = 185 nM T76369 D02HQS 19377173 Ki = 370 nM T76369 D02JVI 44387731 IC50 = 20 nM T76369 D02TLP 11363 Ki = 5270 nM T76369 D03HZT 89076 Ki = 1650 nM T76369 D03NTQ 24951319 IC50 = 5000 nM T76369 D03TPH 87203 Ki = 1220 nM T76369 D03WOU 3274712 Ki = 255 nM T76369 D03XIY 24951160 IC50 = 2000 nM T76369 D04AXR 96047 Ki = 8250 nM T76369 D04CDV 44428829 Ki = 190 nM T76369 D04EXR 251908 Ki = 890 nM T76369 D04PMA 15353606 IC50 = 70 nM T76369 D04UEN 44455866 IC50 = 5.5 nM T76369 D05AVX 60983 Ki = 16900 nM T76369 D05EMT 22574258 Ki = 260 nM T76369 D05EYA 18946 Ki = 1.6 nM T76369 D05LTW 22574224 Ki = 34.7 nM T76369 D05PNO 4135273 Ki = 130 nM T76369 D05VUC 19971657 Ki = 990 nM T76369 D05XRY 2752926 Ki = 2980 nM T76369 D05ZCX 44435802 Ki = 150 nM T76369 D06FFD 96430 Ki = 0.029 nM T76369 D06GYH 16745302 Ki = 260 nM T76369 D06MNW 44285344 IC50 = 9000 nM T76369 D06VGD 6724 Ki = 31 nM T76369 D06VSA 11991809 IC50 = 300 nM T76369 D07CFJ 589576 Ki = 17500 nM T76369 D07EDG 1901244 Ki = 31 nM T76369 D07GOA 11150976 IC50 = 3 nM T76369 D07MSJ 11441196 IC50 = 30000 nM T76369 D08AOG 90571 Ki = 15300 nM T76369 D08UOB 44428840 Ki = 140 nM T76369 D08YHD 9878121 IC50 = 0.5 nM T76369 D09GVB 10427006 IC50 = 600 nM T76369 D09LSR 11437501 Ki = 73.5 nM T76369 D0AW4P 10868634 Ki = 3130 nM T76369 D0B0KP 9977214 IC50 = 500 nM T76369 D0B1BQ 157730 IC50 = 4600 nM T76369 D0B1TQ 1810509 Ki = 5530 nM T76369 D0B8YX 75511 Ki = 125 nM T76369 D0BB2U 2385968 Ki = 524 nM T76369 D0C9AD 277990 Ki = 25 nM T76369 D0C9FO 11991892 IC50 = 2000 nM T76369 D0CH0K 11327355 IC50 = 50000 nM T76369 D0CN8Z 11392969 Ki = 371.54 nM T76369 D0D0BI 8371 Ki = 83.9 nM T76369 D0D2HH 44428834 Ki = 665 nM T76369 D0D7FN 283893 Ki = 213.8 nM T76369 D0D7HU 24950683 IC50 = 80 nM T76369 D0D9GS 24951006 IC50 = 10 nM T76369 D0DW9J 123072 Ki = 229.09 nM T76369 D0E0JC 11279040 IC50 = 700 nM T76369 D0E2IG 44428839 Ki = 320 nM T76369 D0E5CF 185195 Ki = 3.981 nM T76369 D0E5ZP 604575 Ki = 13100 nM T76369 D0EK7H 2734793 Ki = 590 nM T76369 D0F3RN 89801 Ki = 5.4 nM T76369 D0F5VY 94860 Ki = 15.9 nM T76369 D0FO4J 182197 Ki = 5.37 nM T76369 D0G2DQ 4669250 Ki > 100000 nM T76369 D0H5RS 11991808 IC50 = 20 nM T76369 D0I0MR 9840659 IC50 = 4800 nM T76369 D0I7FF 176445 Ki = 2.291 nM T76369 D0JH7C 72810 Ki = 5400 nM T76369 D0JI0H 3542734 Ki = 290 nM T76369 D0K6MH 25147546 IC50 = 30 nM T76369 D0K6OM 44428838 Ki = 300 nM T76369 D0K6PO 316765 Ki = 1.5 nM T76369 D0L1ST 2777298 Ki = 158.49 nM T76369 D0L4MF 44428833 Ki = 170 nM T76369 D0LJ2F 11806279 Ki = 5 nM T76369 D0M2EM 4650 Ki > 100000 nM T76369 D0M2ZD 44428831 Ki = 730 nM T76369 D0M5NR 3794313 Ki = 7690 nM T76369 D0M7SQ 9795477 IC50 = 5 nM T76369 D0M8AR 11154099 IC50 = 50000 nM T76369 D0N0HK 73252 Ki = 5440 nM T76369 D0N1CK 9813810 IC50 = 1 nM T76369 D0N8YZ 2427416 Ki = 18.8 nM T76369 D0N9ZR 1718647 Ki = 16500 nM T76369 D0NJ4G 80771 Ki = 3520 nM T76369 D0O0LU 264734 Ki = 1700 nM T76369 D0P1IK 44428841 Ki = 91.3 nM T76369 D0Q2CR 24950841 IC50 = 25 nM T76369 D0Q2YJ 6763 Ki = 2.5 nM T76369 D0Q3GH 146089 Ki = 4.169 nM T76369 D0S6TW 1845 Ki > 100000 nM T76369 D0SP2O 7054 Ki > 100000 nM T76369 D0T5XC 31494 Ki = 173.78 nM T76369 D0TN0A 10085812 IC50 = 1 nM T76369 D0TP1H 44554615 IC50 = 2500 nM T76369 D0U0BV 44428830 Ki = 1300 nM T76369 D0U3JD 16358 Ki = 5380 nM T76369 D0U8IF 10114 IC50 = 20970 nM T76369 D0U8YV 24951000 IC50 = 0.7 nM T76369 D0UK5A 76996 Ki = 532 nM T76369 D0UT1X 101375 Ki = 18100 nM T76369 D0UZ8R 71043 Ki = 3388.44 nM T76369 D0VQ3O 24799659 IC50 = 30 nM T76369 D0W7NY 11991895 IC50 = 20 nM T76369 D0W9VA 10667 Ki = 930 nM T76369 D0WX6R 3477013 Ki = 570 nM T76369 D0X0ER 344135 Ki = 11400 nM T76369 D0Y0XQ 2779383 Ki > 100000 nM T76369 D0Y6RZ 22574214 Ki = 100 nM T76369 D0Y7FX 8651 Ki = 6.9 nM T76369 D0Z1WQ 76915 Ki = 88.6 nM T76369 D0Z5KQ 8400 Ki = 7210 nM T76369 D0Z6CZ 5139980 Ki = 3020 nM T76369 D0Z7WK 10013998 Ki = 5.248 nM T76369 D0Z8HX 16786802 Ki = 9400 nM T76369 D0ZL6B 3772674 Ki = 16 nM T76369 D0ZR2T 2732752 Ki = 16500 nM T76369 D0ZT5C 44428828 Ki = 480 nM T91323 D05PZB 135398495 IC50 = 10 nM T91323 D07XOV 118598754 IC50 = 131 nM T91323 D0E3TC 44259 IC50 = 30.4 nM T91323 D0T3ME 156422 IC50 > 30000 nM T91323 CP04JC 11666231 IC50 = 12.8 nM T91323 CLS29B 46872626 IC50 > 10000 nM T91323 C8NA4L 53384644 IC50 > 30000 nM T91323 CV63UL 67240318 IC50 > 10000 nM T91323 C0EMZ1 71682213 IC50 = 2100 nM T91323 CQ53SW 71682214 IC50 = 2900 nM T91323 C5N1VZ 102581295 IC50 > 10000 nM T91323 C2B4SW 118714182 IC50 = 630 nM T91323 C4B6PX 118714183 IC50 = 4940 nM T91323 CH91ON 129245363 IC50 = 252 nM T91323 CCF8W2 129261617 IC50 = 25 nM T91323 C9C3XT 134163708 IC50 = 10 nM T91323 CGBZ13 134843302 IC50 = 9600 nM T91323 CJI0G1 135520135 IC50 = 32 nM T91323 CH64ID 136175114 IC50 = 51 nM T91323 C5S8CU 136175115 IC50 = 500 nM T91323 C6X4UA 136175116 IC50 = 780 nM T91323 CJKC57 136175117 IC50 = 250 nM T91323 CJ1NU2 136175118 IC50 = 3000 nM T91323 C3MI1P 136175119 IC50 = 360 nM T91323 CVBM76 136175120 IC50 = 110 nM T91323 C2WP5B 136175121 IC50 = 21 nM T91323 C1TS6F 136175122 IC50 = 120 nM T91323 CB5G4X 136175123 IC50 = 24 nM T91323 C3MK9W 136807986 IC50 > 10000 nM T91323 CSGM03 137210056 IC50 = 12 nM T91323 CW3A2B 137210057 IC50 = 700 nM T91323 C4ZGE1 137210058 IC50 = 1100 nM T91323 CX9RJ6 137210059 IC50 = 460 nM T91323 CBJV93 137210060 IC50 = 320 nM T91323 CPM62S 137210061 IC50 = 360 nM T91323 C6S3UF 137210062 IC50 = 1300 nM T91323 CM0AO9 137210063 IC50 = 24 nM T91323 C4DRX1 137643187 IC50 = 5810 nM T91323 CGW9I0 137656387 IC50 = 1410 nM T91323 C9ISH6 145925685 IC50 = 311 nM T91323 CJB1R5 155511461 IC50 = 15 nM T91323 C2MD1Q 155513187 IC50 > 10000 nM T91323 CHD09S 155543566 IC50 = 30 nM T91323 CO2I4P 155559898 IC50 = 4600 nM T91323 D0GN5Z 5281295 IC50 = 5850 nM T31391 D02EYG 10096344 IC50 = 0.1 nM T31391 D04AIT 5280445 IC50 = 120 nM T31391 D07MGA 72281 IC50 = 280 nM T31391 D0D7LA 4091 IC50 = 29000 nM T31391 D0K8KX 5280343 IC50 = 32730 nM T31391 D0K9MY 11243969 Ki = 0.6 nM T31391 D0L3DK 6918537 Ki = 3 nM T31391 D0N5HJ 5462501 IC50 > 100000 nM T31391 D0NI0C 21704 IC50 = 62 nM T31391 D0NJ5H 11450633 IC50 = 2.7 nM T31391 D0RA5Q 72172 IC50 > 100 ug.mL-1 T31391 D0T8XB 44513473 IC50 = 3.8 nM T31391 D0U2JP 4369359 IC50 = 3.5 nM T31391 D0Y7LD 222284 IC50 = 28840 nM T31391 D04XIO 11253490 IC50 = 23 nM T31391 D05LPW 25022354 IC50 = 0.9 nM T31391 D07EPV 11949652 IC50 = 0.37 nM T31391 D07HZG 11516136 IC50 = 11.3 nM T31391 D0FQ2U 6918572 Ki = 0.18 nM T31391 D0L4FS 5280961 IC50 = 480 nM T31391 D0M3XR 46209133 Ki = 0.8 nM T31391 D0N6SO 15983988 IC50 = 4 nM T31391 D0R9HL 11077541 IC50 = 3.5 nM T31391 D0R9YR 64971 IC50 = 55820 nM T31391 D0U2BH 65064 IC50 = 10210 nM T31391 D0U3EP 445154 IC50 = 0.6 nM T31391 D02LNB 22387295 IC50 = 12 nM T31391 D04MAZ 71731606 IC50 = 0.4 nM T31391 D05FMP 66561557 IC50 > 100000 nM T31391 D07JHU 71667377 IC50 > 100000 nM T31391 D0C6NX 73356493 IC50 > 100000 nM T31391 D0K2ZQ 57378228 IC50 = 0.42 nM T31391 D0QX2U 71667229 IC50 > 100000 nM T31391 D00FYF 9796290 IC50 = 22 nM T31391 D01XGX 178060 IC50 > 100000 nM T31391 D08PUW 64982 IC50 = 225000 nM T31391 D0A1NU 16049769 Ki = 1 nM T31391 D0F3TI 11673176 Ki = 1.8 nM T31391 D0Q4YP 11996845 IC50 = 5.3 nM T31391 D0T2IQ 443600 IC50 > 100 ug.mL-1 T31391 CR40US 18844 IC50 = 7 nM T31391 CT2EY7 56877 IC50 > 100000 nM T31391 CL1Y4H 68247 IC50 = 1410 nM T31391 CBP13T 69512 IC50 = 1410 nM T31391 C0V9WL 73324 IC50 > 100 ug.mL-1 T31391 CHAI28 83489 IC50 = 10360 nM T31391 C8EQ1Z 92855 IC50 = 35600 nM T31391 CP1JX4 124031 IC50 = 23.4 ug.mL-1 T31391 C15AMW 158341 IC50 = 14130 nM T31391 CB9Q1L 168182 IC50 = 65690 nM T31391 C6JM7L 182750 IC50 > 100 ug.mL-1 T31391 CV0J8H 182751 IC50 > 100 ug.mL-1 T31391 CGT6C5 276114 IC50 > 100 ug.mL-1 T31391 C7HME8 439246 IC50 = 240 nM T31391 CT2S6P 441667 IC50 = 420 nM T31391 CPKO72 448436 IC50 = 0.1 nM T31391 CP3EL4 454740 IC50 = 3350 nM T31391 C0GD3A 454742 IC50 = 890 nM T31391 C0TYO2 477693 IC50 = 19.8 ug.mL-1 T31391 C7G3CT 477696 IC50 > 100 ug.mL-1 T31391 C8P2LC 485077 IC50 = 56230 nM T31391 CG3C4U 489605 IC50 = 25000 nM T31391 CSJ38Y 679638 IC50 = 3900 nM T31391 CPEY84 688304 IC50 > 100000 nM T31391 C4TRL6 721814 IC50 > 337500 nM T31391 CO3KZ2 741570 IC50 > 100 ug.mL-1 T31391 C18XUS 978607 IC50 = 2800 nM T31391 C0L7TD 1235479 IC50 = 81 ug.mL-1 T31391 C2HQJ7 2302144 IC50 > 100 ug.mL-1 T31391 C30WIA 2750782 IC50 > 100000 nM T31391 CJW0G1 2854000 IC50 = 4000 nM T31391 CT2CQ8 3021908 IC50 = 21000 nM T31391 CX08LH 3081017 IC50 > 100000 nM T31391 CAZ25S 3318661 IC50 > 1000000 nM T31391 CQ0G4F 5281406 IC50 = 87100 nM T31391 C1DW0R 5316300 IC50 = 38430 nM T31391 CAU3O8 5317238 IC50 = 87720 nM T31391 CFB0N1 5318591 IC50 = 26920 nM T31391 CL6J0E 5320287 IC50 = 41690 nM T31391 CQP43H 5360349 IC50 = 5 nM T31391 CS5BG1 5494385 IC50 = 23 nM T31391 CDG53K 5494422 IC50 = 90 nM T31391 CT0E7G 6293081 IC50 = 33110 nM T31391 CE98OF 6451150 IC50 = 21.88 nM T31391 CPUF51 6918418 IC50 = 5700 nM T31391 C4RE5F 7020797 IC50 = 21000 nM T31391 C48BSO 7614279 IC50 = 26100 nM T31391 C37RIP 9655981 IC50 = 3440 nM T31391 C14VRG 9794073 IC50 = 3900 nM T31391 CQT36A 9794235 IC50 = 1700 nM T31391 CXEQ40 9795464 IC50 = 64 nM T31391 CMVO26 9795469 IC50 = 21 nM T31391 CBG8M2 9796291 IC50 = 1170 nM T31391 CSA6V9 9796352 Ki = 218 nM T31391 C7KR1T 9799867 IC50 = 4 nM T31391 CNJ0Z3 9800721 Ki = 2 nM T31391 C75RIB 9801978 IC50 = 7 nM T31391 C5F7DH 9815545 IC50 = 2 nM T31391 CUNB40 9817010 IC50 = 247000 nM T31391 C1I5JZ 9819537 IC50 = 298 nM T31391 CDP16K 9821063 IC50 = 17000 nM T31391 C8CR0Z 9821205 IC50 = 0.13 nM T31391 CKR9Y5 9823963 IC50 = 13 nM T31391 C8EK7G 9835053 IC50 = 3700 nM T31391 CW5EZ7 9835382 IC50 = 1600 nM T31391 CDY12G 9835472 IC50 = 3100 nM T31391 CV87XC 9835734 Ki = 154 nM T31391 CAHB35 9836210 IC50 = 922 nM T31391 CU2B0F 9838664 IC50 = 110 nM T31391 C62DNH 9843297 IC50 = 27 nM T31391 CUD46C 9855673 IC50 = 188000 nM T31391 CO2YQ4 9858442 IC50 = 69 nM T31391 C8XO1Z 9859008 Ki = 18 nM T31391 CNYI42 9859384 IC50 = 0.6 nM T31391 C2DMP6 9861924 IC50 > 100 ug.mL-1 T31391 CK0BS5 9864687 IC50 = 36 nM T31391 C5CZ6J 9865563 Ki = 53 nM T31391 CF3I8A 9865779 IC50 = 4.6 nM T31391 CR9AW7 9870934 IC50 = 23 nM T31391 CQN2L1 9882325 IC50 = 63 nM T31391 CZUQ34 9883487 IC50 = 460 nM T31391 C2TV9M 9884543 IC50 = 0.064 nM T31391 CBI2C9 9885607 IC50 = 82 nM T31391 CFMG63 9886974 IC50 = 12 ug.mL-1 T31391 CBW37X 9903629 IC50 = 466 nM T31391 C4T1CX 9904675 IC50 = 491 nM T31391 CU0I4K 9907074 IC50 = 270 nM T31391 CMGX12 9920733 IC50 = 23100 nM T31391 C4EC8A 9924995 IC50 = 610 nM T31391 C1S5VM 9927481 IC50 = 436 nM T31391 C6T0RU 9928326 IC50 = 360 nM T31391 C8Y5UK 9939534 IC50 = 23 nM T31391 CFH1V2 9942336 IC50 > 1000000 nM T31391 C28XTC 9942425 Ki = 2000 nM T31391 CZ1S9O 9942554 IC50 = 0.3 nM T31391 CZMT26 9947730 IC50 = 166 nM T31391 C2KW8I 9951445 IC50 = 1.8 nM T31391 CLR78W 9952894 IC50 = 88 nM T31391 CQ8J7T 9953181 IC50 = 59 nM T31391 C8OX9T 9964212 IC50 = 50400 nM T31391 C8THS1 9970277 IC50 = 64000 nM T31391 C1A3YN 9972358 IC50 = 2300 nM T31391 CH39FT 9973732 IC50 = 2000 nM T31391 C9EZ1X 9978478 IC50 = 2.2 nM T31391 CT6XQ2 9983092 IC50 = 1.4 nM T31391 C18ZXU 9990413 IC50 > 1000000 nM T31391 C1NB0Q 9992723 Ki = 79 nM T31391 C5Q6BJ 9995375 IC50 > 100 ug.mL-1 T31391 C17BCF 10003476 IC50 = 1 nM T31391 CN8XI3 10006926 IC50 = 1 nM T31391 CVG9I2 10012350 IC50 > 1000000 nM T31391 C7IB1W 10014222 Ki = 8 nM T31391 C4KT7I 10014539 IC50 > 1000000 nM T31391 CQ7G2R 10018887 IC50 = 1100 nM T31391 CV85MG 10019118 IC50 = 196000 nM T31391 CN0T5A 10019492 IC50 = 7400 nM T31391 C78NMY 10026124 IC50 = 234 nM T31391 CWQ21K 10038196 Ki = 96 nM T31391 CSZ75E 10046311 IC50 = 71 nM T31391 CRG1N0 10058240 IC50 >> 1000000 nM T31391 CYMG54 10058520 Ki = 210 nM T31391 C64ZDU 10059633 IC50 = 545000 nM T31391 CYH3C6 10061400 IC50 > 100 ug.mL-1 T31391 CV7SK8 10064801 IC50 = 57800 nM T31391 CI1Q6X 10081481 IC50 > 500000 nM T31391 CHC82B 10083376 IC50 > 1000000 nM T31391 CSHQ57 10084828 IC50 > 1000000 nM T31391 CB9J1F 10086451 IC50 = 16 nM T31391 C06KTL 10087724 IC50 > 1000000 nM T31391 C97FIB 10087948 IC50 = 245 nM T31391 C83ZDL 10096130 IC50 = 22 nM T31391 C8P3UC 10106636 Ki = 24 nM T31391 C5U0ON 10107122 IC50 = 3.3 nM T31391 C3K2MO 10109454 IC50 = 0.18 nM T31391 C7A3ZJ 10111068 Ki = 79 nM T31391 CKP5D7 10111288 IC50 = 7 nM T31391 CKY4R8 10112957 Ki = 281 nM T31391 CN5BD7 10114895 IC50 = 731 nM T31391 CIU12J 10116290 IC50 = 170 nM T31391 CM19YB 10125495 IC50 = 18000 nM T31391 CQT5Y2 10125644 IC50 = 1400 nM T31391 C10JOC 10125645 IC50 = 2500 nM T31391 CAOF95 10125896 IC50 = 200 nM T31391 C10BSW 10125952 IC50 = 1100 nM T31391 CD20SG 10125953 IC50 = 14000 nM T31391 CT6CG1 10126186 IC50 = 0.2 nM T31391 C0Q7BK 10127057 IC50 = 42 nM T31391 CNC5D4 10130367 Ki = 182 nM T31391 C9ERD7 10130575 IC50 = 22 nM T31391 CBL6T7 10132708 IC50 = 5 nM T31391 CLZF79 10133903 Ki = 12 nM T31391 C2RW5Z 10135822 Ki = 324 nM T31391 C4U3IC 10144962 IC50 = 139 nM T31391 C2H0UF 10149048 Ki = 0.03 nM T31391 C2YUP9 10149491 IC50 = 14000 nM T31391 CUE7K0 10156677 Ki = 112 nM T31391 C4CX1P 10157141 IC50 = 128 nM T31391 CUB1G7 10157334 Ki = 68 nM T31391 C6PZ1U 10160012 Ki = 316 nM T31391 C0L1KV 10162433 Ki = 428 nM T31391 C29RUO 10162817 Ki = 579 nM T31391 CQ3K8W 10164624 IC50 = 1900 nM T31391 C5X4NF 10171676 IC50 = 1000 nM T31391 C98FDL 10172375 IC50 = 0.9 nM T31391 C6SQ0P 10172376 IC50 = 90 nM T31391 CJ3MD2 10172601 IC50 = 100 nM T31391 C2SNQ8 10172681 IC50 = 240 nM T31391 C2KWM9 10172706 IC50 = 3 nM T31391 CXUC74 10173174 IC50 = 130 nM T31391 CKWE80 10176680 Ki = 2.2 nM T31391 C1UAG7 10176937 IC50 = 25 nM T31391 CEM94Y 10178009 IC50 = 539 nM T31391 C6S5OX 10179212 Ki = 29 nM T31391 CF7C3M 10180260 Ki = 45 nM T31391 C4FC2O 10183667 IC50 = 108 nM T31391 C7PWN9 10193213 IC50 = 31000 nM T31391 CWU9N2 10198228 Ki = 3 nM T31391 C05DXJ 10200731 Ki = 302 nM T31391 C6ISW4 10203198 Ki = 309 nM T31391 CD2U3A 10203599 Ki = 63 nM T31391 CQ8N1T 10209865 IC50 = 134 nM T31391 CFP27I 10214732 IC50 = 42000 nM T31391 C0CPY9 10215103 IC50 = 370 nM T31391 CL4T7Z 10215326 IC50 = 270 nM T31391 CLO81K 10215577 IC50 = 1750 nM T31391 C68WBI 10215628 IC50 = 47 nM T31391 CQ0V1C 10219838 IC50 = 39000 nM T31391 CZ9XN0 10220206 IC50 = 170 nM T31391 CBZ3P2 10221723 Ki = 56 nM T31391 CBC45I 10222923 Ki = 1278 nM T31391 CZ92XV 10225547 Ki = 76 nM T31391 CU9W8N 10233525 IC50 = 405 nM T31391 COD64C 10236556 IC50 = 47000 nM T31391 CYCJ68 10236557 IC50 = 1500 nM T31391 C9K3JS 10237877 IC50 = 180 nM T31391 C5P0AO 10238227 IC50 = 113 nM T31391 CTG4S9 10238900 IC50 = 1397 nM T31391 CCS75T 10242745 IC50 > 1000000 nM T31391 CW6PG0 10243173 Ki = 811 nM T31391 C07QCO 10243334 IC50 = 346 nM T31391 C6JS1Y 10245529 IC50 = 42 nM T31391 C0A9OY 10249393 IC50 = 30 nM T31391 CZ90LD 10250452 IC50 = 12 nM T31391 CU8C5K 10254918 IC50 = 5 nM T31391 C17HUN 10255762 IC50 = 8.4 nM T31391 C6ER9U 10269517 IC50 = 50 nM T31391 CQ07AR 10270647 Ki = 33 nM T31391 C9BPX2 10270831 IC50 = 280 nM T31391 CD0P5E 10271196 Ki = 530 nM T31391 CQ36IM 10272290 Ki = 24 nM T31391 C6M4SQ 10286219 IC50 = 1500 nM T31391 CAPB18 10286460 IC50 = 200 nM T31391 CZHS09 10286494 IC50 = 10000 nM T31391 CHWJ15 10286977 IC50 = 0.2 nM T31391 CT6FG8 10287141 IC50 = 340 nM T31391 C7AQS6 10287238 IC50 = 3 nM T31391 CHO8E7 10296151 Ki = 1 nM T31391 CC63ZN 10296260 IC50 = 864 nM T31391 CA7Q8J 10298482 Ki = 65 nM T31391 CY3LK8 10300368 Ki = 310 nM T31391 C9FZ2O 10304081 IC50 = 225 nM T31391 C8J3NA 10304145 IC50 = 44 nM T31391 C7US0V 10304855 IC50 = 114 nM T31391 CJDY62 10306170 IC50 = 14 nM T31391 C5AXF1 10308325 IC50 = 20000 nM T31391 CEGV15 10308355 IC50 = 40000 nM T31391 CNX7Q1 10308853 IC50 = 920 nM T31391 CTZN24 10309295 IC50 = 350 nM T31391 CQYE24 10309373 IC50 = 53 nM T31391 C3FB4T 10310021 IC50 = 91 nM T31391 CY6N9I 10318743 IC50 = 9.6 nM T31391 CF1S8U 10320144 IC50 = 4 nM T31391 C08UHI 10320529 IC50 = 117000 nM T31391 CC2TP8 10321088 IC50 = 5 nM T31391 CNV4R3 10324641 IC50 = 5.8 nM T31391 C0JD8Z 10333136 IC50 = 16 ug.mL-1 T31391 CIAV18 10333629 IC50 >> 1000000 nM T31391 CL72FC 10334538 IC50 > 1000000 nM T31391 C4UTO9 10336929 IC50 = 44 nM T31391 CM6Y1B 10339570 Ki = 5 nM T31391 CXP16T 10340933 IC50 = 15000 nM T31391 C1AEN6 10341846 IC50 > 125000 nM T31391 CEZ95L 10342016 IC50 = 58 nM T31391 CKZT43 10353699 IC50 = 518000 nM T31391 CU6LC2 10355512 IC50 = 104 nM T31391 CR0QC5 10367502 IC50 = 3 nM T31391 CP4M2R 10375745 IC50 = 80 nM T31391 CW70CV 10376453 IC50 >> 1000000 nM T31391 C7UO3L 10376704 Ki = 25 nM T31391 CK07VX 10376940 IC50 = 217000 nM T31391 CK8T4C 10381531 IC50 = 14.1 ug.mL-1 T31391 C79UAO 10381586 IC50 > 100 ug.mL-1 T31391 CQ7J2Z 10383508 IC50 = 15 nM T31391 C2GT0H 10384474 IC50 = 80 nM T31391 CY5M4R 10388027 IC50 = 26 nM T31391 CHZ85I 10393133 IC50 = 4800 nM T31391 CLI51Z 10398371 IC50 > 1000000 nM T31391 C29MEL 10399628 Ki = 22 nM T31391 C2EPA5 10401083 IC50 = 635 nM T31391 C6GWB8 10401570 IC50 > 100 ug.mL-1 T31391 C8NAX7 10403949 IC50 > 500000 nM T31391 CE0AS5 10405951 IC50 = 9 nM T31391 C7R6TZ 10406789 IC50 = 100 nM T31391 CVK1G5 10412922 IC50 = 13 nM T31391 CTK71I 10415171 IC50 = 400 nM T31391 C92DAJ 10415172 IC50 = 5600 nM T31391 C7F8SB 10420127 IC50 = 612 nM T31391 C7YIE3 10423532 Ki = 90 nM T31391 C1O2RY 10426457 IC50 = 11.5 nM T31391 C80ZBS 10429788 IC50 = 71 nM T31391 CUS9F6 10432611 IC50 = 13 nM T31391 C6GHF1 10433039 IC50 = 45 nM T31391 CWCA76 10439426 IC50 = 0.48 nM T31391 CAF71Y 10443207 IC50 = 247000 nM T31391 C4BKD9 10445283 Ki = 959 nM T31391 CO59EL 10450114 IC50 = 6.6 nM T31391 CCTY29 10451878 IC50 = 50 nM T31391 C4OC6P 10455620 IC50 = 175 nM T31391 C1WKE4 10455621 IC50 = 100 nM T31391 CHP37D 10456407 IC50 = 142000 nM T31391 C03IBO 10467163 Ki = 3800 nM T31391 CLV58Q 10468265 IC50 >> 1000000 nM T31391 CH1DG5 10478099 IC50 = 92 nM T31391 CL3H9I 10491923 IC50 > 100 ug.mL-1 T31391 CJ2RK6 10492044 IC50 > 100 ug.mL-1 T31391 CF46MR 10515590 IC50 = 70 nM T31391 C30TAX 10538170 IC50 = 95 nM T31391 CN4BI1 10564514 IC50 = 32 nM T31391 C8KLC3 10584166 IC50 = 11 nM T31391 CK3IW4 10584272 IC50 = 3500 nM T31391 C0KTQ5 10607253 IC50 = 50400 nM T31391 C38IDQ 10608000 IC50 = 250 nM T31391 C4PJ7H 10656779 Ki = 2150 nM T31391 C3YS4K 10659346 IC50 > 100 ug.mL-1 T31391 CN5KG9 10661540 IC50 = 12.8 ug.mL-1 T31391 CH6S5L 10704521 IC50 = 60 nM T31391 CXE71J 10750510 IC50 = 30000 nM T31391 CHA8X6 10751333 IC50 = 94000 nM T31391 CYLO09 10774283 IC50 = 52000 nM T31391 C1LSP2 10779050 IC50 > 100 ug.mL-1 T31391 CL26WQ 10780092 IC50 = 286000 nM T31391 C2KDY6 10798619 IC50 = 374000 nM T31391 C1WG0P 10798659 IC50 = 0.3 nM T31391 C1ZJ4I 10799226 IC50 = 107000 nM T31391 CJKX61 10821833 IC50 = 67000 nM T31391 C7BLJ1 10821834 IC50 > 1000000 nM T31391 CHC1X4 10824414 IC50 = 63 nM T31391 C3E8ID 10845163 IC50 = 15000 nM T31391 CK9SB4 10845727 IC50 = 93000 nM T31391 CCR8J7 10848386 IC50 = 17000 nM T31391 C04XQH 10850290 IC50 > 100 ug.mL-1 T31391 C1QL5M 10858831 IC50 > 1000000 nM T31391 C6QH7S 10860092 IC50 = 18600 nM T31391 C6WGA4 10861905 IC50 = 10 nM T31391 CJ39DG 10872395 IC50 > 500000 nM T31391 CS1LP6 10879478 IC50 = 24200 nM T31391 C3UGO0 10879937 IC50 = 53 nM T31391 C2QEW3 10883432 IC50 = 296 nM T31391 C4A5BM 10902702 IC50 = 598 nM T31391 C6ERS7 10904132 IC50 = 23 nM T31391 CVI2T1 10911918 IC50 = 103000 nM T31391 C42NLJ 10912330 IC50 = 7000 nM T31391 CV46YZ 10912691 IC50 = 33 nM T31391 CG9Q1Y 10923589 IC50 = 133 nM T31391 C9BL6G 10926029 IC50 = 70 nM T31391 CLA05J 10932707 Ki = 10 nM T31391 CPG58B 10943400 IC50 = 475 nM T31391 C6HNK4 10947008 IC50 = 7 nM T31391 CTWI82 10950467 IC50 = 149 nM T31391 CYP97B 10958030 IC50 = 17 nM T31391 CF60BW 10966961 IC50 = 26 nM T31391 CY9CW2 10969177 IC50 = 8 nM T31391 CW63DG 10980018 IC50 = 434000 nM T31391 C63VGB 10993665 IC50 = 64 nM T31391 CM5E1A 11000330 IC50 = 52600 nM T31391 CBFE09 11015514 IC50 = 183 nM T31391 CT9I8W 11020125 IC50 = 9610 nM T31391 CWR9G6 11023706 IC50 = 477000 nM T31391 CX1KF2 11024849 IC50 = 14 nM T31391 CA2OR9 11025044 IC50 = 228 nM T31391 CZ94WH 11025199 IC50 > 500000 nM T31391 C4MD5V 11037154 IC50 > 1000000 nM T31391 CH4TD3 11037548 IC50 = 326000 nM T31391 C0O8HF 11045633 IC50 = 29 nM T31391 CEPQ46 11053284 IC50 = 266 nM T31391 CTMK05 11056962 IC50 = 83 nM T31391 C42WCR 11065479 IC50 > 1000000 nM T31391 C9CYS1 11067211 IC50 = 931000 nM T31391 C9S8AG 11068388 IC50 = 16000 nM T31391 C0FWU4 11069462 IC50 = 22 nM T31391 CVJ81D 11075465 IC50 = 282 nM T31391 CNA61F 11076103 IC50 = 305 nM T31391 C60JXQ 11079321 IC50 > 1000000 nM T31391 C2N6MH 11084500 IC50 = 444 nM T31391 CX07LO 11085063 IC50 = 261 nM T31391 CSRO28 11089704 IC50 = 18 nM T31391 CS48RN 11098969 IC50 = 3000 nM T31391 COAR21 11101478 IC50 = 12000 nM T31391 CMO61N 11109983 IC50 = 338 nM T31391 C10CQP 11112644 IC50 = 62 nM T31391 CA4N0B 11117606 Ki = 11 nM T31391 C9GXD6 11117990 IC50 > 500000 nM T31391 C6QL3H 11122260 IC50 > 1000000 nM T31391 C1X8SI 11127914 IC50 = 398 nM T31391 CF41JX 11127915 IC50 = 105 nM T31391 CJB52P 11129932 IC50 = 3 nM T31391 CWDY68 11138020 IC50 = 192 nM T31391 C26ODF 11150893 IC50 > 500000 nM T31391 CXT8Y2 11151568 IC50 = 6 nM T31391 C4HBU9 11153488 IC50 = 30 nM T31391 CJ7E0N 11163434 IC50 = 0.13 nM T31391 CE94RO 11164254 IC50 = 9.3 nM T31391 C7HRW0 11164704 IC50 = 5 nM T31391 C82GSQ 11165177 IC50 = 77 nM T31391 CSB2T9 11166406 IC50 > 125000 nM T31391 CXR12G 11173505 Ki = 49 nM T31391 CX10UC 11173801 IC50 = 5.6 nM T31391 C5U1FY 11176598 IC50 = 830 nM T31391 CN3D5C 11180149 Ki = 0.59 nM T31391 CJS94B 11187292 IC50 = 5.6 nM T31391 C2ME1R 11187389 Ki = 8.9 nM T31391 CG49PR 11187940 Ki = 1.6 nM T31391 C9HKB7 11188314 IC50 = 23 nM T31391 C5E7VQ 11198004 IC50 = 20 nM T31391 CO9QM2 11198569 IC50 > 100000 nM T31391 CF1LD8 11199808 Ki = 0.4 nM T31391 C40SYQ 11200151 Ki = 8 nM T31391 C68XFD 11205761 IC50 > 1000000 nM T31391 C3BXS4 11206225 Ki = 14500 nM T31391 CMBT59 11207320 IC50 > 250000 nM T31391 CR60FN 11209195 IC50 = 17000 nM T31391 CW8FL2 11209569 IC50 = 301000 nM T31391 CJB87Z 11210511 IC50 = 9.7 nM T31391 C2PN1R 11211023 IC50 = 19 nM T31391 CH87RA 11211119 IC50 = 3.6 nM T31391 CHIZ26 11218348 IC50 = 6.3 nM T31391 C6VKT5 11219158 IC50 = 3700 nM T31391 CK5W4F 11220098 Ki = 143 nM T31391 CXAR72 11220471 IC50 = 250000 nM T31391 CSN6U7 11220682 IC50 = 18 nM T31391 CEUD41 11222126 IC50 = 2.6 nM T31391 CU3BG5 11222807 IC50 = 27 nM T31391 CJ2M8G 11222935 Ki = 1.4 nM T31391 C71YJO 11223701 Ki = 0.9 nM T31391 CK1UE7 11229192 IC50 = 188000 nM T31391 C35JSU 11229576 IC50 = 151000 nM T31391 C3X9SY 11229581 IC50 = 148000 nM T31391 CHX25W 11232123 IC50 = 345000 nM T31391 C0JD5Q 11232605 IC50 = 179000 nM T31391 CYL67P 11232890 Ki = 0.85 nM T31391 CR3PJ9 11233253 IC50 = 8 nM T31391 CVL7H4 11233695 IC50 = 30 nM T31391 C3UA7X 11234761 IC50 = 12 nM T31391 C32ZGY 11234800 IC50 = 3 nM T31391 CBES80 11235729 IC50 = 23 nM T31391 C5AB7G 11236208 IC50 = 1.49 nM T31391 C5CZH3 11242300 IC50 = 2130 nM T31391 CUS5G2 11243728 IC50 = 56000 nM T31391 CH82RJ 11244267 IC50 > 1000000 nM T31391 CDLT06 11245133 IC50 = 63 nM T31391 CQ6C5F 11246131 IC50 = 23 nM T31391 C4VQ0N 11246214 IC50 = 5 nM T31391 C67YUV 11253949 Ki = 3.9 nM T31391 CLJ7A1 11255193 IC50 = 417000 nM T31391 CR6N9B 11256457 IC50 = 430 nM T31391 C8M4XU 11256492 IC50 = 35 nM T31391 C2YS9G 11256520 IC50 = 5 nM T31391 C43HPD 11258527 IC50 = 990 nM T31391 C61KZW 11266019 IC50 = 496000 nM T31391 CN2O0L 11268786 IC50 = 4 nM T31391 CKL1A8 11268930 Ki = 0.93 nM T31391 CHO56W 11269281 IC50 = 570 nM T31391 CM0YI7 11269397 Ki = 0.96 nM T31391 C5IY0L 11269712 IC50 = 95000 nM T31391 CM1A5F 11270889 IC50 = 2.77 nM T31391 CR46GY 11277009 IC50 > 1000000 nM T31391 C17TLH 11277905 IC50 = 43 nM T31391 CXFV02 11278425 Ki = 3.5 nM T31391 CUB62P 11278798 IC50 = 4 nM T31391 CB5SD1 11280296 IC50 = 12 nM T31391 CUK58N 11281626 Ki = 0.4 nM T31391 CL5SH2 11281817 IC50 = 21 nM T31391 C0RWV3 11282205 IC50 = 7400 nM T31391 CWNT74 11283294 IC50 = 25 nM T31391 CUM48L 11288538 IC50 = 1.8 nM T31391 C0U2MV 11289193 IC50 = 205000 nM T31391 CO59DU 11289695 IC50 = 6.5 nM T31391 CTC0P9 11289792 IC50 = 148000 nM T31391 CM85DX 11291335 IC50 = 7800 nM T31391 C1YH5K 11291901 IC50 = 36 nM T31391 CCDX51 11292489 Ki = 3.8 nM T31391 CPD0L4 11292861 Ki = 0.35 nM T31391 CSH2N3 11294846 IC50 = 3 nM T31391 C51QAB 11300739 IC50 = 418000 nM T31391 CZV8P2 11300763 Ki = 10 nM T31391 CAL43D 11302841 IC50 = 13 nM T31391 C1TZY0 11302974 Ki = 42 nM T31391 CAW02M 11303089 IC50 = 14 nM T31391 CDZ79G 11304224 IC50 = 240 nM T31391 C2SOA8 11306467 IC50 = 71 nM T31391 CEJ32C 11306468 IC50 = 71 nM T31391 C06NLF 11309656 IC50 = 190000 nM T31391 C8I1QE 11310450 IC50 = 500000 nM T31391 C47GSV 11310499 IC50 = 23000 nM T31391 CP9LQ0 11312069 IC50 = 278000 nM T31391 CG8SA2 11312331 IC50 = 13 nM T31391 C4GUX3 11312733 IC50 > 500000 nM T31391 CMPH23 11313182 IC50 = 13 nM T31391 CEZ27P 11314348 Ki = 0.6 nM T31391 CM28RS 11314596 IC50 = 890 nM T31391 CL72NR 11314959 Ki = 0.45 nM T31391 CT6MF7 11316670 IC50 = 3 nM T31391 CTG12Q 11321743 IC50 = 23100 nM T31391 C9XYK1 11325183 IC50 = 6.2 nM T31391 CS8OH7 11326271 IC50 = 430 nM T31391 CK6G2V 11335782 Ki = 270 nM T31391 C43RXS 11337326 IC50 = 22 nM T31391 C38ADT 11346439 IC50 = 125000 nM T31391 C5SR4K 11346707 IC50 = 350 nM T31391 C9SJ0O 11347777 Ki = 607 nM T31391 CM4CT0 11348315 IC50 = 10 nM T31391 CM5E2A 11349317 IC50 = 57 nM T31391 C35GXU 11350142 Ki = 10 nM T31391 CNB7G8 11356095 IC50 = 39000 nM T31391 C24QLP 11356421 IC50 = 1000000 nM T31391 C1WOH9 11359214 IC50 > 500000 nM T31391 CK2T6J 11359671 IC50 = 17 nM T31391 CUH3S7 11360493 IC50 = 20 nM T31391 CQ9TJ5 11360810 IC50 = 3.7 nM T31391 CZ93VH 11361944 IC50 = 6 nM T31391 CKP0G9 11362130 IC50 = 34 nM T31391 CZ37IN 11372458 IC50 = 192000 nM T31391 CCNX41 11372959 IC50 = 540 nM T31391 CMZ1S9 11373129 IC50 = 6 nM T31391 CW3QZ7 11374531 IC50 = 19.4 nM T31391 C30JEU 11381416 IC50 = 69 nM T31391 C9FN7U 11381726 IC50 > 500000 nM T31391 CQ0MC7 11383372 IC50 = 200 nM T31391 CH74XT 11383468 IC50 > 500000 nM T31391 CE3O6K 11386357 IC50 = 14 nM T31391 CML13R 11389441 Ki = 7000 nM T31391 CH35IZ 11392716 IC50 = 14 nM T31391 CF01WK 11392988 Ki = 2.9 nM T31391 CL9HN3 11395030 Ki = 2 nM T31391 CD5A7Z 11395141 Ki = 10 nM T31391 CR9EB8 11396245 IC50 = 5 nM T31391 CEZS68 11403720 Ki = 28 nM T31391 CSR53F 11404106 IC50 = 186000 nM T31391 C0X6EK 11404881 Ki = 0.72 nM T31391 CI40EH 11405274 Ki = 57 nM T31391 C50PNA 11405365 Ki = 7.1 nM T31391 C3QZD5 11406220 Ki = 5.5 nM T31391 CTW02K 11406276 Ki = 0.67 nM T31391 CV1E7C 11406559 IC50 = 109 nM T31391 C3S8BD 11415118 IC50 = 5.6 nM T31391 C9AW7O 11416338 IC50 = 5 nM T31391 C0RIS4 11417008 IC50 = 15.1 nM T31391 CW8K3F 11417567 IC50 = 6.8 nM T31391 C2ZT0L 11418204 IC50 = 8 nM T31391 CRZ5F1 11418876 IC50 = 27 nM T31391 CFD62G 11419146 IC50 = 6 nM T31391 CPY7B2 11424308 Ki = 26 nM T31391 C3AZ7K 11426348 IC50 = 15 nM T31391 CB5C1T 11428334 Ki = 12 nM T31391 CY15PU 11429829 Ki = 0.83 nM T31391 CFTC85 11432169 IC50 = 29 nM T31391 C27ITV 11436930 IC50 = 250000 nM T31391 CLF89Y 11437087 IC50 > 1000000 nM T31391 CH39KX 11437726 IC50 = 188000 nM T31391 C82ENX 11439333 IC50 = 7 nM T31391 CRW3G4 11440163 IC50 = 10 nM T31391 CN9ZA8 11441300 IC50 = 68 nM T31391 CH09SE 11447824 IC50 > 1000000 nM T31391 CPNU92 11448828 IC50 = 4.9 nM T31391 CUG51Q 11449442 IC50 = 132000 nM T31391 C9RZC1 11450265 IC50 = 70000 nM T31391 CW27UK 11450266 IC50 = 500000 nM T31391 CZ68MT 11451290 IC50 = 8 nM T31391 CY0JG1 11451461 Ki = 1.6 nM T31391 C0DT1O 11451712 Ki = 7.4 nM T31391 CX5Y7J 11451739 Ki = 10 nM T31391 C6P2BR 11452943 Ki = 0.62 nM T31391 C6US2X 11461807 IC50 = 8 nM T31391 CV71FH 11464036 IC50 = 8 nM T31391 C1M9UX 11469862 Ki = 2.2 nM T31391 CWO06L 11471453 IC50 = 10 nM T31391 C7TOQ4 11472776 IC50 > 500000 nM T31391 CO7T4W 11473127 IC50 > 500000 nM T31391 C53RWU 11474019 IC50 = 266000 nM T31391 C6WT7P 11474308 Ki = 25 nM T31391 C5TQP7 11474372 Ki = 31 nM T31391 CE5A4M 11475797 IC50 = 34.3 nM T31391 C7JWD3 11476287 IC50 = 18 nM T31391 CS4H7X 11481506 Ki = 5.2 nM T31391 C6U9KB 11484559 IC50 = 4 nM T31391 C4G9AM 11484758 IC50 = 510 nM T31391 CPL64M 11486126 Ki = 21 nM T31391 CTD0S4 11486251 Ki = 0.98 nM T31391 CNMA97 11487118 IC50 = 128 nM T31391 CBV79P 11487883 Ki = 0.62 nM T31391 CEHI82 11493140 IC50 > 3000 nM T31391 C06RUA 11493219 IC50 = 64 nM T31391 C3MPY0 11493220 IC50 = 955 nM T31391 CDT16S 11493492 Ki = 28 nM T31391 CUTS18 11494449 IC50 = 2800 nM T31391 C50YHW 11494571 IC50 = 31300 nM T31391 C9PRY1 11494684 IC50 = 811 nM T31391 CJD30Y 11495704 IC50 = 2.3 nM T31391 CGA6Q4 11500119 IC50 = 4000 nM T31391 CAH5Z6 11500899 IC50 = 91 nM T31391 C2D9AT 11500939 Ki = 103 nM T31391 CKWZ03 11501743 IC50 = 80 nM T31391 CH7VS5 11505454 IC50 = 28 nM T31391 CBM01H 11507111 IC50 = 1600 nM T31391 CW38YC 11507527 IC50 = 89 nM T31391 C3XAT0 11507559 IC50 = 687 nM T31391 C62RBF 11507639 IC50 = 261 nM T31391 CF2S9Q 11507721 IC50 > 30000 nM T31391 C30JDP 11508177 IC50 = 1070 nM T31391 CLH62G 11508839 IC50 = 19 nM T31391 CM8QB3 11510166 Ki = 93 nM T31391 CQDM72 11514208 IC50 = 1000 nM T31391 C04OAE 11514331 IC50 = 1110 nM T31391 C7CLT9 11515196 IC50 = 118 nM T31391 CA3FS5 11515240 IC50 = 123 nM T31391 C15UQK 11515912 IC50 = 428 nM T31391 CO95FZ 11516000 IC50 = 1160 nM T31391 C0XVU3 11516085 IC50 = 7.6 nM T31391 C2S8BH 11516511 Ki = 14 nM T31391 CH5A7Q 11518007 IC50 = 2.5 nM T31391 C91OHR 11522044 IC50 > 3000 nM T31391 CJM1L9 11522376 IC50 = 62 nM T31391 C31ZBJ 11522467 IC50 = 689 nM T31391 C2TCM8 11523077 IC50 = 6.6 nM T31391 CY96CU 11523396 IC50 = 14800 nM T31391 CDCI64 11524392 IC50 = 14 nM T31391 C8KB4F 11524437 Ki = 612 nM T31391 CMYN65 11526865 IC50 = 150 nM T31391 C0O3XD 11527019 IC50 = 19 nM T31391 CWH3S0 11529375 IC50 = 52 nM T31391 CMN4Y5 11529427 IC50 = 1220 nM T31391 COL08I 11529539 IC50 = 97 nM T31391 CQ56DV 11529688 IC50 = 257 nM T31391 CXA53K 11529948 IC50 = 208 nM T31391 C10LHK 11531002 IC50 = 371 nM T31391 CV1N6Z 11531612 IC50 = 17 nM T31391 CZFI65 11531704 Ki = 30 nM T31391 C1B8JN 11532057 Ki > 10000 nM T31391 CZ35WN 11533932 IC50 = 13 nM T31391 C63DBH 11537823 Ki = 44 nM T31391 COXK41 11537890 Ki = 137 nM T31391 CKM89Z 11538673 IC50 = 22 nM T31391 CFXG35 11538686 IC50 = 13400 nM T31391 CMD6H8 11538715 IC50 = 5.8 nM T31391 CK36XC 11538961 Ki = 18 nM T31391 CG7I8Z 11538992 IC50 = 21 nM T31391 CPR71X 11540951 IC50 = 2.7 nM T31391 C98GDW 11541277 IC50 = 61 nM T31391 CBR9K8 11541314 IC50 = 7.5 nM T31391 CC5M2E 11544575 IC50 = 69 nM T31391 C1HV5Q 11544965 IC50 = 702 nM T31391 CVT52Y 11545508 IC50 = 30 nM T31391 C6KBN4 11546261 Ki = 2.2 nM T31391 CJIX61 11547698 IC50 = 9.9 nM T31391 C5AR6V 11550675 IC50 = 201 nM T31391 C9I5GV 11551088 IC50 = 26 nM T31391 C5NC3J 11551710 Ki = 21 nM T31391 CY3RK7 11551987 IC50 = 102 nM T31391 C6SA9R 11552616 IC50 = 25600 nM T31391 C2DJ6Y 11552953 Ki = 27 nM T31391 CA16WP 11554165 IC50 = 4.8 nM T31391 CCFP45 11558852 IC50 = 205 nM T31391 CV74GT 11559033 Ki = 143 nM T31391 C85EQW 11559371 IC50 = 50 nM T31391 CDK7I5 11559922 Ki = 0.4 nM T31391 CIZ52M 11561317 Ki = 11 nM T31391 CJF19H 11564906 IC50 = 663 nM T31391 CTE30Z 11565791 IC50 = 164 nM T31391 CL4D9A 11565911 IC50 = 66 nM T31391 CMN2K0 11566106 IC50 = 564 nM T31391 CI5W4Y 11566450 IC50 = 106 nM T31391 CLU15X 11566865 IC50 = 454 nM T31391 C4QG9W 11567318 Ki = 1310 nM T31391 CR37GC 11567606 Ki = 2.9 nM T31391 CAR0J5 11567905 IC50 = 24 nM T31391 CR4I1P 11568333 Ki = 4.4 nM T31391 CL41DG 11569450 Ki = 4.6 nM T31391 CY0A7J 11570138 IC50 = 4.3 nM T31391 CW4LO8 11572237 IC50 = 40000 nM T31391 CH76QT 11572962 IC50 = 8 nM T31391 C8G7UP 11573204 Ki = 49 nM T31391 CHL5Y0 11573374 IC50 = 875 nM T31391 C6F4OE 11573417 IC50 = 132 nM T31391 CAE39I 11573427 IC50 = 84 nM T31391 CCR9Q2 11574031 IC50 = 317 nM T31391 C25SEL 11574694 IC50 = 29 nM T31391 CE03TL 11574811 Ki = 28 nM T31391 CQU80H 11576569 IC50 = 55 nM T31391 C7P0NT 11576820 Ki = 54 nM T31391 CW94NS 11577331 IC50 = 8 nM T31391 CQ86GI 11577431 IC50 = 4.1 nM T31391 CJV39M 11579395 Ki = 377 nM T31391 CW31KG 11579932 IC50 = 61 nM T31391 C0T9NU 11580126 IC50 > 3000 nM T31391 C7BJK9 11580332 IC50 > 30000 nM T31391 C7EA6G 11580446 IC50 > 30000 nM T31391 CVG3B6 11580945 IC50 = 447 nM T31391 CCR0D7 11581247 IC50 = 83 nM T31391 CYT4Z1 11581458 IC50 = 49 nM T31391 CA4XU3 11581644 IC50 = 210 nM T31391 C9J1NO 11581694 IC50 = 24 nM T31391 CS6X0E 11581890 IC50 = 128 nM T31391 CAZL49 11584650 IC50 = 13 nM T31391 CUS2H6 11587911 IC50 > 3000 nM T31391 COH9V8 11589872 IC50 = 2.8 nM T31391 C5JYV7 11591936 IC50 = 8 nM T31391 CSCW37 11592154 IC50 = 2.6 nM T31391 CDE3P6 11594121 IC50 = 33 nM T31391 C3NT1E 11594414 IC50 = 160 nM T31391 CA51WQ 11595401 IC50 = 33 nM T31391 CI0E4X 11595565 Ki = 2.2 nM T31391 CO0QJ8 11596007 Ki = 1530 nM T31391 CE8M3K 11596123 Ki = 67 nM T31391 C9MXO0 11596219 IC50 = 116 nM T31391 CW48NY 11596451 Ki = 6.7 nM T31391 CMUV42 11596607 IC50 = 5.2 nM T31391 CSW3M9 11597271 IC50 = 6.9 nM T31391 C9SC1G 11602166 IC50 = 9400 nM T31391 CY4W0X 11602707 IC50 = 11 nM T31391 CHM2N0 11602713 Ki = 317 nM T31391 C9CM7N 11603627 IC50 = 18 nM T31391 CBE6K8 11603637 Ki = 22 nM T31391 CPXV24 11603996 IC50 = 17 nM T31391 C9N2EZ 11604004 Ki = 6.8 nM T31391 CGAF90 11604063 IC50 = 3059 nM T31391 CL4NM7 11604454 IC50 = 676 nM T31391 C0S2RQ 11605368 IC50 = 4.6 nM T31391 C15DLO 11608317 IC50 > 33000 nM T31391 C5V1XM 11608625 IC50 > 3000 nM T31391 C9JZM7 11608919 IC50 > 3000 nM T31391 C6I0XG 11609419 IC50 = 1500 nM T31391 COF62W 11611325 Ki = 9 nM T31391 CAOP57 11612570 IC50 = 715 nM T31391 CQL5S8 11613750 IC50 = 6.2 nM T31391 CZ91WO 11616288 IC50 = 630 nM T31391 C27JCR 11616775 IC50 = 13600 nM T31391 C6MO9K 11616857 IC50 = 651 nM T31391 CD3YU1 11616861 IC50 = 74 nM T31391 CEX4O6 11617338 IC50 = 54 nM T31391 C7KS2Q 11617492 IC50 = 600 nM T31391 C40ZJT 11619382 IC50 = 73 nM T31391 C2APG7 11623550 IC50 = 72 nM T31391 CR8XO2 11623606 IC50 = 59 nM T31391 C7QC6U 11623777 Ki = 1280 nM T31391 C17XSP 11623929 Ki = 8.3 nM T31391 CPSN73 11624012 Ki = 20 nM T31391 CH2JP9 11624034 IC50 > 30000 nM T31391 CDZ72J 11624893 IC50 = 1108 nM T31391 CRY2D5 11625412 Ki = 50 nM T31391 C7YKC0 11628195 IC50 = 22 nM T31391 C5AKH1 11630368 IC50 = 2000 nM T31391 CYR61O 11630666 IC50 = 320 nM T31391 CV17GF 11631125 IC50 = 66 nM T31391 CA1J8U 11631434 IC50 = 3300 nM T31391 CH3WM8 11632024 IC50 = 8400 nM T31391 CSO1D6 11632159 Ki = 43 nM T31391 CZT57X 11632256 IC50 = 52 nM T31391 C8Y3FM 11632315 IC50 = 29 nM T31391 CM1DR9 11632375 Ki = 22 nM T31391 C09KAV 11632502 IC50 = 17 nM T31391 C7SP9Y 11634778 Ki > 3000 nM T31391 CR6NM8 11638575 Ki = 33 nM T31391 CM6QE9 11638687 IC50 > 3000 nM T31391 CHLA97 11638762 Ki = 241 nM T31391 CRA0H5 11639131 Ki = 550 nM T31391 C0M1HR 11640120 IC50 = 4.8 nM T31391 C5P3NB 11644467 IC50 = 56 nM T31391 C3RZO9 11645337 IC50 = 452 nM T31391 CQO8U6 11648011 Ki > 10000 nM T31391 CXG1B4 11649741 IC50 = 6.3 nM T31391 CO2YH1 11652954 Ki = 764 nM T31391 C1Y2DC 11652956 Ki = 867 nM T31391 CZBD50 11653749 Ki = 96 nM T31391 C94OMG 11654093 Ki = 18 nM T31391 C8AU5P 11654528 Ki = 38 nM T31391 CUX2M0 11654810 Ki = 7.2 nM T31391 C52ION 11655271 Ki = 19 nM T31391 CT4W8K 11659101 IC50 = 790 nM T31391 C7M6ZY 11659120 IC50 = 45200 nM T31391 CR8Z6I 11659133 IC50 > 30000 nM T31391 CZFV81 11661472 IC50 = 260 nM T31391 CI8EF3 11666622 IC50 > 3000 nM T31391 CN3WA7 11668525 IC50 > 3000 nM T31391 CE91WR 11669357 IC50 = 20 nM T31391 C43OVS 11673852 IC50 = 96 nM T31391 CCBS09 11674180 Ki = 64 nM T31391 CH1KG5 11674534 IC50 = 57 nM T31391 CTNO72 11674721 IC50 = 4.6 nM T31391 C2G6RP 11675637 Ki = 75 nM T31391 CI1ED9 11676224 IC50 = 150 nM T31391 C3Y7EL 11678025 IC50 = 5.2 nM T31391 C1A7NS 11680394 IC50 = 98 nM T31391 C5BD4Q 11680960 Ki = 12 nM T31391 CV0XW8 11680991 IC50 = 298 nM T31391 CFX6Z9 11681207 IC50 = 32 nM T31391 CNF1M4 11681778 IC50 = 50 nM T31391 C2K9XG 11688776 IC50 = 10 nM T31391 C0IWC9 11689866 IC50 = 651 nM T31391 CA69TN 11690566 IC50 = 77 nM T31391 C8UYQ5 11690713 IC50 = 2500 nM T31391 CC9O1L 11692537 Ki = 0.27 nM T31391 CEAN27 11694995 Ki = 1610 nM T31391 CBW6A1 11695523 IC50 = 6300 nM T31391 C79ECL 11695535 IC50 = 3236 nM T31391 C45QIU 11695818 IC50 = 2800 nM T31391 C7DCV9 11696495 Ki = 438 nM T31391 C6JPE0 11696912 Ki = 495 nM T31391 CRU2Q1 11697286 Ki = 5.6 nM T31391 C2WK1Z 11697387 Ki = 20 nM T31391 C1KCR6 11702577 IC50 = 15000 nM T31391 C2F6BA 11702880 Ki = 15 nM T31391 C8SI4E 11702902 IC50 = 119 nM T31391 C0Q3IL 11703158 IC50 = 784 nM T31391 C8IQA2 11703413 IC50 = 90 nM T31391 CUJ07L 11703663 Ki = 720 nM T31391 CJP1U8 11703749 IC50 = 1.5 nM T31391 C2X5GC 11704411 Ki = 9 nM T31391 C6YHK3 11704412 Ki = 24 nM T31391 CFO63Q 11704578 IC50 = 527 nM T31391 C1MGA4 11705197 Ki = 2.7 nM T31391 C8LA3E 11705712 Ki = 76 nM T31391 CU8LZ4 11705859 IC50 = 1418 nM T31391 CUC0Z3 11708771 IC50 = 400 nM T31391 CZF5D9 11708829 IC50 = 63 nM T31391 CNG85M 11710587 Ki = 8.9 nM T31391 CK4I6J 11710700 Ki = 6 nM T31391 C0CG5R 11710963 IC50 = 42 nM T31391 C04OMI 11711314 Ki = 113 nM T31391 C8VC2D 11711413 Ki = 33 nM T31391 C8KD6N 11711414 Ki = 163 nM T31391 C0U7QC 11715518 IC50 = 105 nM T31391 C34BEP 11716483 Ki = 12 nM T31391 CMI90R 11716843 Ki = 3.4 nM T31391 CCR80L 11717090 IC50 = 116 nM T31391 CZS71R 11717268 IC50 = 369 nM T31391 C1XD5I 11718004 Ki = 113 nM T31391 C1M7PL 11718857 Ki = 30 nM T31391 CY1S3Q 11719625 IC50 = 2.8 nM T31391 C0UJ7G 11719823 IC50 = 910 nM T31391 CIEJ54 11720809 IC50 = 5.3 nM T31391 CHA7Z9 11722557 IC50 = 119 nM T31391 CIOY84 11723708 IC50 = 21.3 ug.mL-1 T31391 C6VG7O 11727562 IC50 = 989 nM T31391 CJ6XR8 11730284 IC50 > 125000 nM T31391 CX9U4G 11731880 IC50 = 503000 nM T31391 C96TGJ 11746838 IC50 = 988 nM T31391 CA2H1U 11747757 IC50 = 163 nM T31391 C3ZPG6 11772582 IC50 = 68 nM T31391 CX84PY 11772583 IC50 = 590 nM T31391 C1P9ZM 11776124 IC50 > 1000000 nM T31391 C6JY7V 11776638 Ki = 8 nM T31391 CS0WM6 11778955 IC50 = 320 nM T31391 C3MX2I 11781105 IC50 = 24 nM T31391 CO73AL 11784400 IC50 = 15000 nM T31391 CKTJ04 11791651 IC50 = 291 nM T31391 C67TXV 11791652 IC50 = 109000 nM T31391 C1P2AI 11809137 IC50 = 102 nM T31391 C6ET2R 11817181 IC50 = 43500 nM T31391 CK24XY 11819467 IC50 > 1000000 nM T31391 C19HAP 11825584 IC50 = 89000 nM T31391 CN79VL 11840913 Ki = 6.7 nM T31391 CSOC43 11840914 Ki = 0.82 nM T31391 CE6V2H 11840916 Ki = 3.8 nM T31391 C42BOS 11854299 IC50 = 56.9 nM T31391 C2FN7G 11854301 IC50 = 53.4 nM T31391 CQ0O5A 11952574 IC50 = 120 nM T31391 CQIB43 11957945 IC50 = 82 nM T31391 CTQI92 11974546 Ki = 45 nM T31391 C5BZW6 11998979 Ki = 140 nM T31391 CXHC16 11999086 Ki = 240 nM T31391 CU3HD8 11999088 Ki = 190 nM T31391 CLI17Z 11999090 Ki = 220 nM T31391 C8U5NY 11999093 Ki = 15 nM T31391 CBZ03A 11999206 Ki = 76 nM T31391 C2TAJ9 11999207 Ki = 200 nM T31391 C3E4ZB 11999208 Ki = 34 nM T31391 C6DK9R 11999211 Ki = 35 nM T31391 CQSP03 12043866 IC50 = 207000 nM T31391 C35DEQ 12043867 IC50 = 3400 nM T31391 C1P3MJ 12043868 IC50 = 18000 nM T31391 C7NRQ3 12043869 IC50 = 731000 nM T31391 CAI8E7 12043870 IC50 = 51400 nM T31391 C21PAF 12069363 IC50 = 0.6 nM T31391 CQY50P 12742483 IC50 = 250000 nM T31391 C9RA7N 13478499 Ki = 160000 nM T31391 CYV1F7 13784835 IC50 > 100 ug.mL-1 T31391 C1GF7B 13939278 IC50 = 750 nM T31391 C94FPE 14434173 IC50 > 100 ug.mL-1 T31391 CR8H4L 14978092 IC50 = 200 nM T31391 CJAE28 15036410 IC50 = 118000 nM T31391 C6BHJ9 15101668 IC50 > 1000000 nM T31391 C29IHT 15337406 IC50 = 16000 nM T31391 CNM5V2 15940321 IC50 = 32360 nM T31391 C2ZMH8 15948988 IC50 = 25.4 nM T31391 C13JIX 15949418 IC50 = 0.67 nM T31391 C49NUJ 15949507 IC50 = 5.3 nM T31391 CPD3V1 15949508 IC50 = 0.5 nM T31391 CU4P5X 15950383 Ki = 3 nM T31391 C16XRI 15950384 Ki = 51.5 nM T31391 CUMR27 15950385 Ki = 11 nM T31391 C69RAY 15950386 Ki = 9 nM T31391 CM63YP 15950387 Ki = 29 nM T31391 CH8F7W 15950388 Ki = 4 nM T31391 C0L4SH 15950456 Ki = 14 nM T31391 C8G7OJ 15950457 Ki = 12 nM T31391 C8FU1V 15950462 Ki = 29 nM T31391 C9KJ6D 15950538 Ki = 2.7 nM T31391 C3C6PM 15950539 Ki = 9 nM T31391 C4S7AB 15950540 Ki = 4 nM T31391 C2HGJ0 15950541 Ki = 16 nM T31391 C3U1VO 15950542 Ki = 9 nM T31391 CKX8M6 15950615 Ki = 4 nM T31391 CC0M2X 15951427 Ki = 8 nM T31391 CF3PX0 15951428 Ki = 30 nM T31391 CWTX01 15951429 Ki = 12 nM T31391 C3LQD9 15951431 Ki = 18 nM T31391 C8M0FT 15951543 IC50 = 27 nM T31391 CI3DB4 15951636 IC50 > 20000 nM T31391 C3SM4T 15951642 IC50 > 100000 nM T31391 C8QRV9 15951839 Ki = 38400 nM T31391 CMNT83 15951928 Ki = 608000 nM T31391 CL1E6O 15953860 IC50 = 17 nM T31391 CG2E3Z 15991577 IC50 = 84 nM T31391 CLG2Q1 16035093 IC50 = 24 nM T31391 CMUG74 16035094 IC50 = 25 nM T31391 CYPG43 16040279 Ki = 3.2 nM T31391 C13-MAR 16040457 IC50 > 100000 nM T31391 C0YQ9A 16046127 IC50 = 325000 nM T31391 C75ZNE 16058650 Ki = 4 nM T31391 C28IRJ 16064807 IC50 = 17 nM T31391 C4LJH3 16064808 IC50 = 24 nM T31391 CVIC15 16064809 IC50 = 11 nM T31391 CS7DQ3 16090844 Ki = 3 nM T31391 C8CVG9 16090856 Ki = 1.3 nM T31391 CB6WK0 16121107 Ki = 170000 nM T31391 CZQ8O9 16121199 Ki = 100000 nM T31391 C5Q9BH 16122596 IC50 = 16 nM T31391 CU3GB5 16126742 IC50 = 4.8 nM T31391 CUQT90 16202787 Ki = 12 nM T31391 CHUX72 16202788 Ki = 3.8 nM T31391 C8D2RM 16203032 Ki = 1400 nM T31391 CW0JF5 16203033 Ki = 17 nM T31391 C5F6DE 16203034 Ki = 590 nM T31391 C0LJA8 16203036 Ki = 105 nM T31391 CC20IT 16203037 Ki = 4 nM T31391 CW6AC3 16203151 Ki = 6 nM T31391 C5BE1I 16204461 Ki = 1600 nM T31391 CWY50B 16204462 Ki = 930 nM T31391 CAQ7S4 16204463 Ki = 440 nM T31391 CCW34I 16204464 Ki = 270 nM T31391 CCWF31 16204465 Ki = 83 nM T31391 C73HLC 16204466 Ki = 24 nM T31391 CA1PV5 16216352 IC50 > 33000 nM T31391 CD9MQ6 16223559 IC50 = 245 nM T31391 CQ7G8T 16223560 IC50 = 1.7 nM T31391 CN24YP 16223762 IC50 = 984 nM T31391 CF37TH 16226604 IC50 = 84 nM T31391 C6ANU2 16226605 IC50 = 109 nM T31391 CFW43X 16658022 IC50 = 5 nM T31391 C6H5VO 16658023 IC50 = 5 nM T31391 CC9W4S 16658024 IC50 = 15 nM T31391 CR51WX 16658101 IC50 = 13 nM T31391 CMLR19 16658102 IC50 = 5 nM T31391 CXN32U 16658103 IC50 = 8 nM T31391 C2XP7B 16658104 IC50 = 4 nM T31391 CD6L7Z 16658105 IC50 = 19 nM T31391 C63NWG 16658243 IC50 < 10 nM T31391 C82ZAL 16658881 IC50 = 460 nM T31391 C24NZK 16658917 Ki = 2.3 nM T31391 C28GEM 16662696 IC50 = 1.1 nM T31391 C53XZP 16721117 Ki = 2 nM T31391 CW62MC 16725327 IC50 = 1.3 nM T31391 C0EV4T 16725905 IC50 = 5 nM T31391 C56LTN 16739329 IC50 = 0.92 nM T31391 CT01PQ 16739331 IC50 = 70 nM T31391 C19UBP 16747699 IC50 = 13 nM T31391 C9JK5Q 16750059 Ki = 5.3 nM T31391 C61RFP 16755651 Ki = 13 nM T31391 C4RK2Q 17591662 IC50 = 94.82 nM T31391 CU05RG 17748274 IC50 = 16 nM T31391 C15TBF 17751406 IC50 = 15000 nM T31391 C5W3VY 17753031 IC50 = 76 nM T31391 CX5F2U 17763521 IC50 > 500000 nM T31391 CQG89Z 17853548 IC50 = 41400 nM T31391 C6L7MA 18391459 IC50 = 2.9 nM T31391 CV4Z6Q 18398587 IC50 = 134900 nM T31391 CP3S0V 18398588 IC50 = 247000 nM T31391 C7GDU9 20038035 IC50 > 100 ug.mL-1 T31391 CC8RN3 20198196 IC50 = 18100 nM T31391 CT42AI 20706081 IC50 = 330 nM T31391 CBZ1E6 21045424 IC50 = 765 nM T31391 C6ZMS8 21054400 Ki = 5 nM T31391 CWB93R 21054485 IC50 = 21 nM T31391 CBY6M2 21919450 IC50 = 142 nM T31391 CH7YL4 21919455 IC50 = 10000 nM T31391 C1PF7M 21919463 IC50 = 2200 nM T31391 C39STQ 21919469 IC50 = 1150 nM T31391 C2OXL1 21919478 IC50 = 13 nM T31391 CY8OJ7 21947630 IC50 = 26 nM T31391 CQ9LB5 21947637 IC50 = 89 nM T31391 CCFX26 21947643 IC50 = 7 nM T31391 C3SXF7 21947646 IC50 = 4 nM T31391 CPES59 21949259 IC50 = 190000 nM T31391 C2W4KV 21949272 IC50 = 67000 nM T31391 CZ9K4Q 22029435 IC50 = 580 nM T31391 C0X4SO 22029457 IC50 = 340 nM T31391 CLK4G6 22029894 IC50 = 1230 nM T31391 C6BME5 22175258 IC50 = 1100 nM T31391 CRA87P 22175262 IC50 = 360 nM T31391 C7E0NG 22175290 IC50 = 2400 nM T31391 C2SD9C 22175298 IC50 = 2400 nM T31391 CQ3EB8 22175361 IC50 = 47 nM T31391 C56RIP 22175474 IC50 = 1900 nM T31391 C28HMT 22175479 IC50 = 1100 nM T31391 CK4NR7 22175497 IC50 = 1200 nM T31391 C2ME4A 22175534 IC50 = 870 nM T31391 C2RM7H 22175568 IC50 = 980 nM T31391 C7X5DS 22175618 IC50 = 3800 nM T31391 CE3LM6 22175639 IC50 = 250 nM T31391 CLUH89 22175659 IC50 = 4000 nM T31391 C4AUK1 22175709 IC50 = 8300 nM T31391 C6KGB8 22175713 IC50 = 220 nM T31391 CBYP16 22175758 IC50 = 250 nM T31391 CB38EC 22176094 IC50 = 1500 nM T31391 CR23XQ 22176165 IC50 = 2400 nM T31391 C8QF7T 22176298 IC50 = 1900 nM T31391 CUND82 22176405 IC50 = 1600 nM T31391 CL68SA 22220623 IC50 = 80000 nM T31391 C2XAR9 22401333 IC50 > 100000 nM T31391 CED47V 22690988 IC50 = 24000 nM T31391 C9VGC8 22691359 IC50 > 100000 nM T31391 C43XCK 22691633 Ki = 5300 nM T31391 C1M2ZS 22691666 IC50 > 100000 nM T31391 CM4SH2 23595882 IC50 = 167000 nM T31391 CP1J3T 23596395 Ki = 14 nM T31391 C8JSI4 23628284 IC50 = 50 nM T31391 CC29GD 23633277 IC50 = 0.5 nM T31391 C1RV7P 23633348 IC50 = 17 nM T31391 CU1LK3 23633350 IC50 = 1.5 nM T31391 CKN67W 23633553 IC50 = 6 nM T31391 CG37EL 23633557 IC50 = 7 nM T31391 C5U3NL 23633697 IC50 = 9 nM T31391 CVC80Z 23633837 IC50 = 10 nM T31391 C8P9GL 23633839 IC50 = 400 nM T31391 C5UVZ9 23634061 IC50 = 60 nM T31391 C5ZF2X 23634210 IC50 = 25 nM T31391 C4KW2T 23634279 IC50 = 4 nM T31391 CVF78O 23634281 IC50 = 4 nM T31391 CA95UP 23634434 IC50 = 8.4 nM T31391 C7FSW5 23634528 IC50 > 36900 nM T31391 CAQ81M 23644660 IC50 = 455 nM T31391 CDPU25 23644665 IC50 = 7360 nM T31391 CCSU21 23645371 IC50 = 27 nM T31391 C5M6UX 23645373 Ki = 470 nM T31391 CFS6P4 23645374 Ki = 20 nM T31391 CAVN39 23645375 Ki = 26 nM T31391 CN0FR1 23645376 Ki = 3.1 nM T31391 CVQ39W 23645377 Ki = 5.3 nM T31391 CQPA42 23645378 Ki = 36 nM T31391 CQ5R2G 23645379 Ki = 360 nM T31391 C32KIA 23645380 Ki = 1160 nM T31391 C6TCN1 23645381 Ki > 12800 nM T31391 CL08ZV 23645382 Ki > 12800 nM T31391 C8P3OQ 23645383 Ki > 12800 nM T31391 C72KLP 23645384 Ki = 980 nM T31391 CNVP26 23645385 Ki = 360 nM T31391 C3OHM9 23645386 Ki = 310 nM T31391 C8TP3W 23645387 Ki = 166 nM T31391 CZXL64 23645388 Ki = 160 nM T31391 C7MAX0 23645389 Ki = 170 nM T31391 C7W6PC 23645390 Ki = 96 nM T31391 CX0VJ4 23645391 Ki = 8900 nM T31391 C4EM3K 23645392 Ki > 12800 nM T31391 CU76EP 23645393 Ki > 12800 nM T31391 CFV07G 23645410 IC50 = 231 nM T31391 CIMG82 23645411 IC50 = 68 nM T31391 C47OZL 23645510 IC50 = 520 nM T31391 C2Q5IK 23645581 IC50 = 48 nM T31391 C3VA0M 23645582 IC50 = 968 nM T31391 C1JAG6 23645622 IC50 = 110 nM T31391 CDL4G9 23645678 Ki = 2.1 nM T31391 CL1DC7 23645680 Ki = 1.8 nM T31391 C23BMA 23645681 IC50 = 170000 nM T31391 C4B9FM 23645685 Ki = 1 nM T31391 CP9GS5 23645686 IC50 = 19700 nM T31391 C6R2LP 23645687 IC50 = 1820 nM T31391 CN7FK3 23645688 IC50 = 12400 nM T31391 CSHX17 23645689 IC50 = 4790 nM T31391 CL8QV6 23645690 IC50 = 4820 nM T31391 C0AU9X 23645691 IC50 = 990 nM T31391 CRM3Y4 23645692 IC50 = 15600 nM T31391 CDM8A2 23645693 IC50 = 3820 nM T31391 CIR1F6 23645694 IC50 = 1790 nM T31391 CK5G6I 23645695 IC50 = 1610 nM T31391 CHS76O 23645696 IC50 = 330 nM T31391 CVP59D 23645697 IC50 = 190 nM T31391 CH13BW 23645698 IC50 = 122 nM T31391 CL0K1T 23645699 IC50 = 520 nM T31391 CB3Z7O 23645700 IC50 = 4590 nM T31391 CNO6Q1 23645702 IC50 = 160 nM T31391 CGMC54 23645703 IC50 = 830 nM T31391 C0V4WR 23645705 IC50 = 43 nM T31391 CY9XW5 23645721 IC50 = 40 nM T31391 C5MO2Q 23645882 Ki = 260 nM T31391 C1UR3L 23645883 Ki = 507 nM T31391 C5EQ1C 23645884 Ki > 10000 nM T31391 CO90SF 23645885 Ki = 212 nM T31391 C85TUY 23645886 Ki = 1311 nM T31391 CBNC76 23645887 Ki = 140 nM T31391 CE1H2R 23645888 Ki = 513 nM T31391 CR7C8Q 23645889 Ki > 10000 nM T31391 CSW5F3 23645890 Ki = 4422 nM T31391 C7E8AI 23645891 Ki > 10000 nM T31391 C8YGE5 23645892 Ki = 399 nM T31391 C31TSP 23645893 Ki > 10000 nM T31391 C87LMT 23645894 Ki > 10000 nM T31391 CX79LQ 23645895 Ki = 74 nM T31391 CON27H 23645896 Ki = 27 nM T31391 CAYT68 23645897 Ki = 673 nM T31391 C5SH6W 23645898 Ki = 37 nM T31391 CDFZ57 23645899 Ki = 188 nM T31391 C5XB6V 23645900 Ki > 10000 nM T31391 CS6WQ4 23645901 Ki = 18 nM T31391 C9AZD2 23645902 Ki = 3 nM T31391 C2O6ML 23645903 Ki = 23 nM T31391 CKM6Y8 23645917 IC50 = 250 nM T31391 C9Y2ZL 23645918 IC50 = 110 nM T31391 C4V6BX 23645919 IC50 = 130 nM T31391 C78PNU 23645920 IC50 = 150 nM T31391 C5YT6S 23645921 IC50 = 180 nM T31391 CELQ89 23645922 IC50 = 150 nM T31391 CGV92H 23645923 IC50 = 350 nM T31391 CJ60EH 23645924 IC50 = 160 nM T31391 CZG70A 23645925 IC50 = 160 nM T31391 CD6V7X 23645926 IC50 = 220 nM T31391 C1TD4J 23645927 IC50 = 300 nM T31391 C71PQU 23645928 IC50 = 270 nM T31391 C8EOB9 23645929 IC50 = 780 nM T31391 C0M1TH 23645930 IC50 = 150 nM T31391 CFHB36 23645931 IC50 = 130 nM T31391 CTG27F 23645932 IC50 = 39 nM T31391 CS2FT5 23645933 IC50 = 72 nM T31391 C98QGK 23645934 IC50 = 160 nM T31391 CS76DY 23645935 IC50 = 130 nM T31391 C91MYK 23645936 IC50 = 85 nM T31391 C3AQC0 23645937 IC50 = 590 nM T31391 C61GTC 23645938 IC50 = 480 nM T31391 C8XF6R 23645939 IC50 = 310 nM T31391 C7IX5B 23645940 IC50 = 360 nM T31391 CP6M3W 23645941 IC50 = 260 nM T31391 CQ75XK 23645942 IC50 = 380 nM T31391 C8T7GY 23645943 IC50 = 130 nM T31391 C25ZXC 23645944 IC50 = 290 nM T31391 C4A3NI 23645945 IC50 = 180 nM T31391 C9Y1BP 23646016 IC50 = 73 nM T31391 CL8DY2 23646017 IC50 = 73 nM T31391 CT6Q1R 23646018 IC50 = 72 nM T31391 C8VS1X 23646019 IC50 = 144 nM T31391 CL4BX5 23646020 IC50 = 4130 nM T31391 CZ24WC 23646021 IC50 = 1957 nM T31391 C98VYW 23646022 IC50 = 2587 nM T31391 CCL17M 23646023 IC50 = 228 nM T31391 CT16HE 23646024 IC50 = 129 nM T31391 CAL8T5 23646025 IC50 = 63 nM T31391 CVSH12 23646026 IC50 = 274 nM T31391 C15HJB 23646027 IC50 > 100000 nM T31391 CBUM54 23646029 IC50 > 100000 nM T31391 C32ZNH 23646030 IC50 = 31000 nM T31391 CE8L2I 23646031 Ki = 64 nM T31391 C8SIU2 23646032 IC50 > 100000 nM T31391 C7L6JR 23646033 IC50 > 100000 nM T31391 CJ9ZL3 23646080 IC50 > 1000000 nM T31391 C0S2UB 23646081 IC50 > 1000000 nM T31391 CQ3KF6 23646082 IC50 > 1000000 nM T31391 CZ9P0Q 23646083 IC50 > 1000000 nM T31391 CFPN10 23646084 IC50 > 1000000 nM T31391 C0NV1B 23646085 IC50 > 1000000 nM T31391 CSW9T1 23646086 IC50 > 250000 nM T31391 CH72RP 23646087 IC50 > 1000000 nM T31391 CH5Y2F 23646088 IC50 > 500000 nM T31391 CJ47OR 23646089 IC50 > 250000 nM T31391 CRT2B0 23646090 IC50 > 250000 nM T31391 C7JXN0 23646091 IC50 > 1000000 nM T31391 C4K1NE 23646092 IC50 > 250000 nM T31391 CJV2K1 23646093 IC50 > 250000 nM T31391 C51BSR 23646094 IC50 > 250000 nM T31391 C2WDG4 23646095 IC50 > 125000 nM T31391 CB2ZT7 23646096 IC50 > 1000000 nM T31391 COF57U 23646097 IC50 > 1000000 nM T31391 CU26YP 23646098 IC50 > 250000 nM T31391 CM37ZS 23646100 IC50 > 1000000 nM T31391 C4SV2J 23646101 IC50 > 1000000 nM T31391 CX68KV 23646102 IC50 > 1000000 nM T31391 CZ28UC 23646142 Ki = 62 nM T31391 CLA15H 23646143 Ki = 4 nM T31391 C0EK5I 23646441 IC50 = 7.2 nM T31391 CF1TP9 23646442 IC50 = 160 nM T31391 CZA78Q 23646443 IC50 = 89 nM T31391 C5VP2I 23646444 IC50 = 14 nM T31391 C9PW1E 23646445 IC50 = 150 nM T31391 CAI0B5 23646446 IC50 = 2300 nM T31391 C4XM2W 23646447 IC50 = 67000 nM T31391 CUZ0D8 23646448 IC50 = 142 nM T31391 C7PE0S 23646449 IC50 = 16 nM T31391 COT87G 23646450 IC50 = 0.91 nM T31391 CF2J9Q 23646451 IC50 = 0.49 nM T31391 CVHU93 23646508 Ki = 9 nM T31391 CJLP47 23646509 Ki = 10 nM T31391 C7P5TW 23646510 Ki = 22 nM T31391 C61FRE 23646511 Ki = 1200 nM T31391 C4EG5D 23646512 Ki = 11 nM T31391 CN47RA 23646513 Ki = 29 nM T31391 CDM3J0 23646514 Ki = 25 nM T31391 CW0J6X 23646515 Ki = 57 nM T31391 CS6L8X 23646516 Ki = 300 nM T31391 COPD36 23646517 Ki = 260 nM T31391 CWT7X1 23646518 Ki = 450 nM T31391 C5GQ7J 23646519 Ki = 11 nM T31391 C0E8SM 23647079 IC50 = 280 nM T31391 CA6X5F 23647080 IC50 = 39 nM T31391 CP2W3B 23647081 IC50 = 3800 nM T31391 CS8O6P 23647082 IC50 = 820 nM T31391 CA53BK 23647084 IC50 = 110 nM T31391 CK15XF 23647085 IC50 = 340 nM T31391 CFOA63 23647106 IC50 = 13 nM T31391 CRF32I 23647107 IC50 = 5 nM T31391 CFTW63 23647114 IC50 = 20.7 nM T31391 C0BQ2D 23647115 IC50 = 11.6 nM T31391 CLO1Y2 23647116 IC50 = 69.9 nM T31391 CSJ78F 23647117 IC50 = 9 nM T31391 CDE9L7 23647118 IC50 = 11.5 nM T31391 CZF25M 23647119 IC50 = 15.1 nM T31391 CW5U3C 23647120 IC50 = 10.5 nM T31391 CWO62C 23647121 IC50 = 19.2 nM T31391 C0X1CK 23647122 IC50 = 8 nM T31391 C7JOV9 23647123 IC50 = 33 nM T31391 C0UT7J 23647124 IC50 = 397 nM T31391 C8P2VJ 23647125 IC50 = 37.3 nM T31391 CQ85KB 23647126 IC50 = 60.3 nM T31391 CRFL12 23647127 IC50 = 24.6 nM T31391 CP3CF0 23647128 IC50 = 143 nM T31391 CJA3M7 23647129 IC50 = 142 nM T31391 C7L3RX 23647130 IC50 = 11 nM T31391 C8UWB7 23647132 IC50 = 29.6 nM T31391 C60MWC 23647133 IC50 = 126 nM T31391 C8TZD5 23647134 IC50 = 2 nM T31391 CBA8N1 23647136 IC50 = 21 nM T31391 CG0U2M 23647137 IC50 = 33 nM T31391 C3TSN4 23647138 IC50 = 37 nM T31391 C6QKM4 23647139 IC50 = 310 nM T31391 CQPN26 23647141 IC50 = 780 nM T31391 C4V5TC 23647142 IC50 = 995 nM T31391 C8TDA5 23647143 IC50 = 1247 nM T31391 CNRH86 23647144 IC50 = 1325 nM T31391 CY19JV 23647145 IC50 = 1460 nM T31391 C39DJX 23647146 IC50 = 1995 nM T31391 C4P2IJ 23647147 IC50 = 2209 nM T31391 CTB09J 23647311 IC50 = 13 nM T31391 CJ6XT7 23647314 IC50 = 18 nM T31391 CVI19F 23653088 IC50 = 3800 nM T31391 CO9GD8 23655077 IC50 = 22 nM T31391 CWVR37 23655298 IC50 > 500000 nM T31391 CPCX60 23655474 IC50 > 1000000 nM T31391 CB1E5P 23655476 IC50 > 500000 nM T31391 CWTD09 23655478 IC50 > 1000000 nM T31391 CLSE92 23655741 IC50 > 40200 nM T31391 CQ53MU 23655742 IC50 > 36900 nM T31391 C4DOR0 23655937 IC50 > 41300 nM T31391 CRA46X 23655938 IC50 > 39100 nM T31391 CW9UR3 23657402 IC50 > 250000 nM T31391 CU18EA 23657547 IC50 > 250000 nM T31391 CVF6E2 23661697 IC50 = 25 nM T31391 CM7C4W 23661708 IC50 = 26 nM T31391 CO6L9F 23661716 IC50 = 1.2 nM T31391 CHR14F 23661718 IC50 = 6 nM T31391 CG8TJ9 23824719 IC50 = 11000 nM T31391 CNP9T1 24180585 IC50 = 37 nM T31391 CO0ZA3 24692381 IC50 = 67000 nM T31391 CR7I3Y 24703639 IC50 > 1000000 nM T31391 CVA72K 24704198 IC50 = 374000 nM T31391 CKWZ51 24710701 IC50 = 360000 nM T31391 CKVQ51 24749924 IC50 = 1 nM T31391 CCW9N3 24749925 IC50 = 4 nM T31391 CXNY61 24749926 IC50 = 4 nM T31391 CZ4BH0 24749927 IC50 = 284 nM T31391 C9X8CK 24750044 IC50 = 5 nM T31391 CK7V6L 24750165 IC50 = 56 nM T31391 C7I4LK 24750278 IC50 = 3 nM T31391 CT21RV 24750279 IC50 = 2 nM T31391 CC6X1F 24750280 IC50 = 88 nM T31391 C5TIP2 24750281 IC50 = 9 nM T31391 C7QSH2 24752844 IC50 = 65 nM T31391 CI0W8A 24755210 IC50 = 1.3 nM T31391 CU7W4F 24768547 IC50 = 0.21 nM T31391 CX8DH1 24769723 IC50 = 1.4 nM T31391 C0H8OB 24776705 IC50 = 116 nM T31391 C24GLZ 24776939 IC50 = 0.18 nM T31391 C6LD2J 24777439 IC50 = 209 nM T31391 CK8EL5 24777568 IC50 = 12 nM T31391 CQ20PV 24777692 IC50 = 88 nM T31391 C1WF3I 24777804 IC50 = 4.3 nM T31391 C50SPA 24784161 IC50 = 123 nM T31391 C29SZR 24784416 IC50 = 90000 nM T31391 C0H8IZ 24784426 IC50 = 116 nM T31391 CO7L6R 24784427 IC50 = 73 nM T31391 C8FQT4 24784664 IC50 > 100000 nM T31391 C69QMZ 24784674 IC50 = 238 nM T31391 CW8LK2 24784675 IC50 = 47 nM T31391 CH1W5N 24784676 IC50 = 140 nM T31391 CJ0ZI7 24784677 IC50 = 251 nM T31391 CIZF59 24784915 IC50 = 72 nM T31391 CKFH56 24784916 IC50 = 195 nM T31391 C5HY0P 24784918 IC50 = 212 nM T31391 CS6HU2 24784925 IC50 = 182 nM T31391 CK6W8S 24784926 IC50 = 45 nM T31391 CUH32V 24785152 IC50 = 305 nM T31391 C2KL7G 24794725 IC50 = 63 nM T31391 CUM03S 24798754 IC50 = 0.12 nM T31391 CZ3ND1 24832041 IC50 = 32 nM T31391 CY9W8O 24860300 IC50 = 1 nM T31391 CKZ25G 24862861 IC50 = 7.5 nM T31391 CFNZ09 24893980 IC50 = 3670 nM T31391 CMK9B7 24894026 IC50 > 100000 nM T31391 CSIK84 24906298 IC50 = 500000 nM T31391 CYL69J 24951732 IC50 = 0.7 nM T31391 CNP3T1 24951733 IC50 = 3.7 nM T31391 CDCP18 24952087 IC50 = 7.3 nM T31391 CIM7S2 24952089 IC50 = 3.5 nM T31391 CX83WL 24963343 IC50 > 100000 nM T31391 CDU69X 24999325 IC50 = 50 nM T31391 CA94RD 24999327 IC50 = 9 nM T31391 CZJ2N6 24999330 IC50 = 24 nM T31391 C9ML5P 24999630 IC50 = 14 nM T31391 C3VU2K 24999632 IC50 = 69 nM T31391 CUO7Q4 24999636 IC50 = 120 nM T31391 CM6AW8 24999638 IC50 = 39 nM T31391 CY90LJ 25014552 IC50 = 2740 nM T31391 CA28YZ 25017799 IC50 = 2.28 nM T31391 C40ONC 25021195 IC50 = 223 nM T31391 C67ZQD 25054021 IC50 = 357 nM T31391 C3SW1V 25054553 IC50 = 64 nM T31391 CH9F2B 25054555 IC50 = 64 nM T31391 CHO68D 25054557 IC50 = 56 nM T31391 C3R9XM 25054809 IC50 = 50 nM T31391 C2D4LI 25054811 IC50 = 3 nM T31391 CHE83A 25054815 IC50 = 13 nM T31391 CXPO63 25054817 IC50 = 68 nM T31391 CA2EK8 25055067 IC50 = 328 nM T31391 C8J9ZG 25055304 IC50 = 80 nM T31391 C51KTQ 25055741 IC50 = 7.4 nM T31391 CI0K2T 25055743 IC50 = 4.3 nM T31391 C1Q6RS 25055745 IC50 = 2.2 nM T31391 CIA48J 25055828 IC50 = 204 nM T31391 CA3N5B 25055836 IC50 = 229 nM T31391 CEDP80 25055999 IC50 = 1.7 nM T31391 C5K3QM 25056001 IC50 = 11 nM T31391 CGX3K8 25056003 IC50 = 17 nM T31391 C6X9PG 25056005 IC50 = 5.2 nM T31391 C8P7VJ 25056091 IC50 = 601 nM T31391 CN83UK 25056093 IC50 = 77 nM T31391 C0LJF5 25056353 IC50 = 6 nM T31391 CS81DK 25056618 IC50 = 112 nM T31391 CQM3U1 25056620 IC50 = 192 nM T31391 C7WEY3 25056875 IC50 = 807 nM T31391 C62UCV 25056881 IC50 = 95 nM T31391 CK7B2E 25057130 IC50 = 102 nM T31391 CQCY54 25057136 IC50 = 25 nM T31391 CM3AU5 25057138 IC50 = 17 nM T31391 CR26DS 25057390 IC50 = 309 nM T31391 C8Q2GP 25057392 IC50 = 175 nM T31391 C9TQ7J 25057396 IC50 = 680 nM T31391 C6KHT4 25057400 IC50 = 1700 nM T31391 C6Q2CM 25057648 IC50 = 88 nM T31391 C1RN5F 25057650 IC50 = 101 nM T31391 CUF2P9 25057652 IC50 = 212 nM T31391 CQHM69 25110577 IC50 = 510 nM T31391 CTS7I5 25110685 IC50 = 3.6 nM T31391 CHTM74 25110898 IC50 = 2500 nM T31391 CBC24W 25110901 IC50 = 8500 nM T31391 CW3GZ6 25112031 IC50 = 710 nM T31391 C76RFD 25112033 IC50 = 2200 nM T31391 CYV1T4 25112035 IC50 = 1900 nM T31391 CW7UD1 25112037 IC50 = 1600 nM T31391 CX9NR5 25112039 IC50 = 3000 nM T31391 CN2MQ8 25112155 IC50 = 770 nM T31391 CO7UE8 25112157 IC50 = 3700 nM T31391 CUIW48 25112159 IC50 = 3100 nM T31391 C6B8CF 25112161 IC50 = 2000 nM T31391 CQ0GY8 25112163 IC50 = 1600 nM T31391 CI71VQ 25112265 IC50 = 8900 nM T31391 CR13HD 25112267 IC50 = 1900 nM T31391 CWE10R 25112269 IC50 = 3600 nM T31391 CK69WG 25112271 IC50 = 1400 nM T31391 C5W8KL 25112273 IC50 = 5900 nM T31391 CXM0N5 25112374 IC50 = 2800 nM T31391 CK16JS 25112376 IC50 = 4300 nM T31391 C9KF5T 25112378 IC50 = 2200 nM T31391 C5O9PU 25112380 IC50 = 2700 nM T31391 C19DPQ 25112382 IC50 = 1400 nM T31391 CYJ2B5 25112487 IC50 = 2700 nM T31391 CUA2K9 25112489 IC50 = 1600 nM T31391 C60EOS 25112491 IC50 = 5600 nM T31391 CV75BU 25112493 IC50 = 1600 nM T31391 CDL2S7 25112495 IC50 = 7400 nM T31391 CF97YP 25112497 IC50 = 1300 nM T31391 CDKE79 25112619 IC50 = 2100 nM T31391 C4TLZ7 25112621 IC50 = 9100 nM T31391 CI3KP5 25112623 IC50 = 690 nM T31391 CF9BO5 25112625 IC50 = 4800 nM T31391 C5QA1K 25112627 IC50 = 2600 nM T31391 C01GPL 25132159 Ki = 8.3 nM T31391 C7IDX9 25132160 IC50 = 0.89 nM T31391 C9VK8W 25132161 Ki = 17 nM T31391 CFZ4V2 25132162 Ki = 3300 nM T31391 CSU0B5 25189891 Ki = 14.4 nM T31391 CA98HO 25203967 IC50 = 2000 nM T31391 CPMN48 28787393 IC50 = 6.29 nM T31391 C9Q2OH 42601533 IC50 = 3850 nM T31391 C0BC9N 42601535 IC50 = 350 nM T31391 C7KN2U 42608447 IC50 = 0.38 nM T31391 C60SVD 42636924 IC50 = 15 nM T31391 C76NLT 42773972 IC50 > 250000 nM T31391 C6LQN3 43181622 IC50 > 1000000 nM T31391 C42OZD 43271345 IC50 = 377000 nM T31391 CK54OM 43650152 IC50 = 229000 nM T31391 CS40ML 44123747 IC50 = 1.1 nM T31391 CSX10M 44138030 IC50 = 4 nM T31391 CQF86D 44182505 IC50 = 13 nM T31391 C3I4TF 44201003 IC50 = 10 nM T31391 CE5B7H 44218404 IC50 = 13 nM T31391 CR8GT4 44218550 IC50 = 15 nM T31391 CBW7D4 44218551 IC50 = 39 nM T31391 CVH08B 44218552 IC50 = 18 nM T31391 CISE95 44218553 IC50 = 27 nM T31391 CLB72R 44218554 IC50 = 14 nM T31391 C2N9VR 44218555 IC50 = 63 nM T31391 CJ6L3S 44218693 IC50 = 29 nM T31391 C97IFE 44218695 IC50 = 32 nM T31391 C50EKW 44250174 IC50 = 9 nM T31391 CRZI12 44266022 IC50 = 14 nM T31391 C9YT6M 44270944 Ki = 1.1 nM T31391 C4MSN1 44285301 IC50 = 7900 nM T31391 CP9YN0 44285888 IC50 = 7000 nM T31391 CT3U1W 44286225 IC50 = 2400 nM T31391 C5UA6S 44286288 IC50 = 103000 nM T31391 CMG71F 44286291 IC50 = 52600 nM T31391 CQ5H8W 44286293 IC50 = 18000 nM T31391 CB6R9L 44286310 IC50 = 948000 nM T31391 C7ZHL3 44286477 IC50 = 277000 nM T31391 CF2H7C 44286480 IC50 = 746000 nM T31391 C7YU4C 44286501 IC50 = 6700 nM T31391 C0HZ5A 44286513 IC50 = 8400 nM T31391 C54LIM 44286562 IC50 = 170000 nM T31391 CH72YN 44286743 IC50 = 31800 nM T31391 C58LKI 44286823 IC50 = 14000 nM T31391 CVQ7K3 44286825 IC50 = 4700 nM T31391 CL3Q2J 44306072 IC50 = 4000 nM T31391 CMC8B9 44306777 IC50 = 44 nM T31391 CF2Q5V 44325514 Ki = 0.5 nM T31391 CE6G4X 44325523 Ki = 450 nM T31391 CI2YN1 44325525 Ki = 260 nM T31391 C29OIF 44325533 Ki = 0.8 nM T31391 CV4QM7 44325534 Ki = 6000 nM T31391 CLDY18 44325535 Ki = 4200 nM T31391 CN46PE 44325540 Ki = 21 nM T31391 CX94HW 44325697 Ki = 5 nM T31391 C1GRJ2 44325719 Ki = 0.41 nM T31391 CN45KP 44325734 Ki = 1.7 nM T31391 C4WTQ7 44326630 IC50 = 109000 nM T31391 C98LVO 44326651 IC50 = 372 nM T31391 C51EOL 44326652 IC50 = 218 nM T31391 C49PEQ 44326772 IC50 = 18700 nM T31391 C8NS4L 44326791 IC50 = 242 nM T31391 CYHE81 44327018 IC50 = 256 nM T31391 CNH8J3 44327071 IC50 = 16 nM T31391 CR3GE1 44327072 IC50 = 15 nM T31391 CSU32T 44327098 IC50 = 377 nM T31391 C0XFT4 44327160 IC50 = 13 nM T31391 CG7K1P 44327192 IC50 = 123 nM T31391 C2RC9I 44328126 IC50 = 14000 nM T31391 CTC40N 44328274 Ki = 47600 nM T31391 C8M0SH 44328300 Ki = 200 nM T31391 C6NZ9C 44328318 IC50 = 213000 nM T31391 C6OHV2 44328319 IC50 > 500000 nM T31391 CA53DN 44330624 IC50 = 13000 nM T31391 C7E1BJ 44330636 IC50 = 68000 nM T31391 C75JRD 44360575 IC50 = 24 nM T31391 CS72FI 44360697 IC50 = 7.5 nM T31391 CKSO92 44360724 IC50 = 26 nM T31391 CYED53 44360725 IC50 = 89 nM T31391 CXEC92 44360726 IC50 = 35 nM T31391 CL7WM8 44360734 IC50 = 64 nM T31391 CA0U8X 44360744 IC50 = 98 nM T31391 C50NME 44360749 IC50 = 94 nM T31391 CKI6W3 44360785 IC50 = 18 nM T31391 CRM9Y7 44360786 IC50 = 24 nM T31391 CXTP74 44360787 IC50 = 2.6 nM T31391 C5MB1D 44360809 IC50 = 46 nM T31391 C29DTA 44360810 IC50 = 190 nM T31391 CPTX82 44360812 IC50 = 2700 nM T31391 C3M8KF 44360910 IC50 = 38 nM T31391 CR7Q9N 44360911 IC50 = 53 nM T31391 CFY7P3 44360924 IC50 = 33 nM T31391 C62HNE 44360925 IC50 = 33 nM T31391 C1H5YG 44360938 IC50 = 21 nM T31391 C6IZ8L 44360955 IC50 = 15 nM T31391 CCJA09 44360967 IC50 = 29 nM T31391 CLMF32 44360976 IC50 = 20 nM T31391 CV1YL5 44360977 IC50 = 17 nM T31391 CY8A9K 44361010 IC50 = 10 nM T31391 C2KWI0 44361074 IC50 = 17 nM T31391 C1Z2FV 44361086 IC50 = 55 nM T31391 C8MJY5 44361216 IC50 = 9 nM T31391 CYK42S 44361230 IC50 = 25 nM T31391 CM3R2T 44364102 IC50 = 250000 nM T31391 CJ0VM6 44364126 IC50 = 3500 nM T31391 C83IUZ 44364133 IC50 = 217000 nM T31391 CJ8N0S 44364172 IC50 > 1000000 nM T31391 C7D2FW 44364210 IC50 = 93000 nM T31391 C8HO2F 44364211 IC50 = 500000 nM T31391 C9IQG4 44364212 IC50 > 1000000 nM T31391 C47NKP 44364213 IC50 = 52000 nM T31391 C6CYU9 44364227 IC50 > 500000 nM T31391 CHLV59 44364231 IC50 > 500000 nM T31391 CZF5N2 44364237 IC50 > 1000000 nM T31391 C7VR0N 44364252 IC50 > 1000000 nM T31391 CTS8U3 44364253 IC50 > 1000000 nM T31391 C0IW9L 44364296 IC50 = 289000 nM T31391 C6FBH7 44364297 IC50 = 81000 nM T31391 C79JMS 44364298 IC50 = 318000 nM T31391 CF2TA0 44364385 IC50 = 151000 nM T31391 C19DCN 44364405 IC50 = 51000 nM T31391 CX5AK7 44364446 IC50 > 500000 nM T31391 C4XIV2 44364456 IC50 > 1000000 nM T31391 C3XN5A 44364457 IC50 = 107000 nM T31391 CKA86J 44364458 IC50 = 500000 nM T31391 C4QON9 44368427 IC50 = 12.8 ug.mL-1 T31391 C8FB1S 44368725 IC50 = 64.4 ug.mL-1 T31391 CE83AK 44368726 IC50 > 100 ug.mL-1 T31391 CW9BG0 44368735 IC50 = 18.7 ug.mL-1 T31391 C37TIM 44368736 IC50 = 15.1 ug.mL-1 T31391 CX8I6C 44381633 IC50 = 550 nM T31391 CW9F3N 44381634 IC50 = 1200 nM T31391 CI39RJ 44381635 IC50 = 210 nM T31391 CLK90J 44381645 IC50 = 95 nM T31391 CT0EO4 44381646 IC50 = 240 nM T31391 CHX2T7 44381647 IC50 = 1100 nM T31391 C6Y4QW 44381687 IC50 = 110 nM T31391 CN96MI 44381721 IC50 = 420 nM T31391 CK4SP1 44381763 IC50 = 480 nM T31391 CI6RT5 44381811 IC50 = 4600 nM T31391 CG1CD7 44381826 IC50 = 110 nM T31391 CL51SX 44381845 IC50 = 660 nM T31391 CXBY42 44381846 IC50 = 230 nM T31391 C5SV9U 44381847 IC50 = 110 nM T31391 CRY5K1 44381848 IC50 = 3900 nM T31391 CRE8J7 44381849 IC50 = 280 nM T31391 CUX2Q9 44381861 IC50 = 220 nM T31391 C92CKY 44381862 IC50 = 130 nM T31391 CIX09S 44381884 IC50 = 46 nM T31391 C3GH0S 44381896 IC50 = 43 nM T31391 C0FQO1 44381899 IC50 = 47 nM T31391 CTRX81 44381910 IC50 = 420 nM T31391 C2XBA5 44381911 IC50 = 170 nM T31391 CBL60E 44381919 IC50 = 250 nM T31391 CARK25 44381928 IC50 = 94 nM T31391 C4LR3K 44381945 IC50 = 270 nM T31391 CQ4VZ3 44381966 IC50 = 440 nM T31391 CDCY49 44381967 IC50 = 670 nM T31391 CT9IN5 44381974 IC50 = 330 nM T31391 C0FQY4 44381979 IC50 = 180 nM T31391 CP7XG9 44382005 IC50 = 180 nM T31391 C6YFP9 44382006 IC50 = 870 nM T31391 CWJ3V5 44382013 IC50 = 1700 nM T31391 CI8O3F 44382065 IC50 = 150 nM T31391 CX2JS7 44382077 IC50 = 72 nM T31391 C38MSH 44382133 IC50 = 110 nM T31391 C8PD7J 44382134 IC50 = 83 nM T31391 C89LXF 44382393 IC50 = 840 nM T31391 CAJ50V 44382443 IC50 = 290 nM T31391 C8ZP1A 44382444 IC50 = 110 nM T31391 CKOD04 44382521 IC50 = 83 nM T31391 CY2C8J 44387751 IC50 > 1000000 nM T31391 CXSU53 44387755 IC50 > 1000000 nM T31391 CALG81 44387756 IC50 > 1000000 nM T31391 CL1M7V 44387758 IC50 > 125000 nM T31391 C6T2MW 44387765 IC50 > 1000000 nM T31391 CA7KI2 44390794 IC50 = 13000 nM T31391 CVD21W 44393563 IC50 = 39640 nM T31391 C24PMT 44393585 IC50 > 100000 nM T31391 CB9WA5 44393586 IC50 = 16480 nM T31391 C7N1GB 44393611 IC50 = 3000 nM T31391 CS51KL 44393656 IC50 = 33000 nM T31391 C7SB1I 44393657 IC50 = 44860 nM T31391 C9JT0N 44393695 IC50 = 46910 nM T31391 CPG38C 44393696 IC50 = 27470 nM T31391 CF6KR8 44393727 IC50 = 51000 nM T31391 C58KPC 44393728 IC50 = 5700 nM T31391 CDH6J1 44393857 IC50 = 200 nM T31391 C2PK9W 44393881 IC50 = 2620 nM T31391 CB6E5I 44393933 IC50 = 80 nM T31391 C08BMZ 44394001 IC50 = 51 nM T31391 C8RA0W 44394023 IC50 = 9400 nM T31391 C3KH1Q 44394024 IC50 = 589 nM T31391 C4QE5X 44394028 IC50 = 143 nM T31391 CPF49E 44394029 IC50 = 155 nM T31391 C8ZA9M 44394031 IC50 = 11000 nM T31391 CS35UP 44394072 IC50 = 2026 nM T31391 CW79MD 44394073 IC50 = 19 nM T31391 CW81MP 44394103 IC50 = 270 nM T31391 C7Y4LZ 44394104 IC50 = 8476 nM T31391 C25SDY 44394118 IC50 = 19000 nM T31391 CU85FA 44394119 IC50 = 30 nM T31391 CJ18AZ 44394135 IC50 = 35000 nM T31391 CTEP50 44394136 IC50 = 36000 nM T31391 C4BO3S 44394155 IC50 = 34 nM T31391 CALF89 44394157 IC50 = 0.1 nM T31391 C4B9OH 44394173 IC50 = 1100 nM T31391 CX75VF 44394180 IC50 = 14860 nM T31391 C85SEO 44394194 IC50 = 2519 nM T31391 CS1Z7X 44394195 IC50 = 2263 nM T31391 C39LZT 44394203 IC50 = 3028 nM T31391 CF6Y8L 44394209 IC50 = 10700 nM T31391 CQ09FB 44394210 IC50 = 1040 nM T31391 CXG8B6 44394238 IC50 = 931 nM T31391 CIJ95E 44394239 IC50 = 981 nM T31391 C3Q5WZ 44394241 IC50 = 3611 nM T31391 CL3EP4 44394242 IC50 = 690 nM T31391 C8U2ZQ 44394244 IC50 = 3279 nM T31391 CZA46H 44394270 IC50 = 2026 nM T31391 CUGH58 44394271 IC50 = 8951 nM T31391 CU7PY3 44394282 IC50 = 7688 nM T31391 C41ITO 44394305 IC50 = 1900 nM T31391 CG53YO 44394349 IC50 = 1552 nM T31391 C59NLA 44394350 IC50 = 1700 nM T31391 C0NSL3 44396153 IC50 = 4 nM T31391 C1VLP6 44399148 IC50 = 252 nM T31391 CIED90 44399244 IC50 = 87 nM T31391 C3PKV8 44399546 IC50 = 97 nM T31391 CEW52I 44400445 IC50 = 0.25 nM T31391 C8UDI1 44400447 IC50 = 0.33 nM T31391 CZ19WH 44400450 IC50 = 6.6 nM T31391 C0MEB2 44400462 IC50 = 1.5 nM T31391 C41SZA 44400473 IC50 = 0.28 nM T31391 C68USM 44400485 IC50 = 0.19 nM T31391 CZ6A8Q 44400504 IC50 = 3 nM T31391 CJD9B5 44400535 IC50 = 5.5 nM T31391 CU8CL1 44400547 IC50 = 6.7 nM T31391 CR87KM 44400555 IC50 = 1.9 nM T31391 CSJU72 44400574 IC50 = 4.6 nM T31391 C6VB2Q 44400588 IC50 = 9.7 nM T31391 C3RAW7 44400625 IC50 = 0.53 nM T31391 CUR51H 44402967 Ki = 504 nM T31391 CZO5J3 44402970 Ki = 1267 nM T31391 CIKW98 44402971 Ki = 61 nM T31391 CP72TO 44402972 Ki = 81 nM T31391 CA8K9B 44403068 Ki = 109 nM T31391 C32LIY 44403069 Ki = 117 nM T31391 CPX1M9 44403336 IC50 = 370 nM T31391 CSEN70 44403337 IC50 = 17000 nM T31391 C0NXE8 44403338 IC50 = 2000 nM T31391 CR53EK 44403354 IC50 = 1200 nM T31391 CRO16Q 44403360 IC50 = 4.5 nM T31391 C0FC7D 44403361 IC50 = 15 nM T31391 C3HFZ7 44403391 IC50 = 130 nM T31391 C3TOY4 44403392 IC50 = 75 nM T31391 CU39LX 44403393 IC50 = 25 nM T31391 CIA8Y3 44403397 IC50 = 27 nM T31391 C6P7NE 44403398 IC50 = 58 nM T31391 CP34SF 44403405 IC50 = 8 nM T31391 C60VBT 44403406 IC50 = 61 nM T31391 C50LWV 44403411 IC50 = 16000 nM T31391 CQ5T4Y 44403412 IC50 = 0.8 nM T31391 CMX9B1 44403416 IC50 = 12 nM T31391 CUKG07 44403417 IC50 = 560 nM T31391 CX29FU 44403421 IC50 = 1600 nM T31391 C2P4CQ 44403422 IC50 = 7.8 nM T31391 CCOA39 44403438 IC50 = 32000 nM T31391 CLYJ80 44403439 IC50 = 810 nM T31391 C4YAH3 44404393 IC50 = 25 nM T31391 C02SYC 44406179 Ki = 225 nM T31391 CU8B3S 44406189 Ki = 46 nM T31391 C1SBD5 44406234 Ki = 115 nM T31391 C5P1RX 44406284 Ki = 40 nM T31391 C0IQO3 44411572 IC50 = 771 nM T31391 C3HXA1 44411573 IC50 > 3000 nM T31391 CW73SO 44411579 IC50 > 3000 nM T31391 CB17FI 44411652 IC50 > 3000 nM T31391 C5WPL4 44411659 IC50 > 3000 nM T31391 C1HCZ6 44411660 IC50 > 3000 nM T31391 C29ZOU 44411665 IC50 > 3000 nM T31391 C9MH4X 44411669 IC50 > 3000 nM T31391 C54RFY 44411670 IC50 > 3000 nM T31391 CE86UP 44411700 IC50 = 237 nM T31391 CR7MX8 44411923 IC50 = 1860 nM T31391 CFP80H 44412105 Ki = 0.41 nM T31391 CZ15VN 44412163 Ki = 2.5 nM T31391 C0HA7I 44412169 Ki = 2900 nM T31391 CGJ17L 44415883 IC50 > 250000 nM T31391 CE0KW2 44415905 IC50 > 100000 nM T31391 CPR49A 44415906 IC50 > 125000 nM T31391 CQ5P2J 44415929 IC50 = 234000 nM T31391 CM2W5X 44415930 IC50 > 125000 nM T31391 COPZ87 44415944 IC50 > 125000 nM T31391 CGLB32 44417381 Ki = 49 nM T31391 C2TP5K 44417385 Ki = 97 nM T31391 CN2F6U 44417389 Ki > 30000 nM T31391 C12HGD 44417391 Ki > 30000 nM T31391 CSG4F8 44417393 Ki = 1 nM T31391 CE7UB0 44418114 IC50 = 0.29 nM T31391 CD9J3S 44418157 IC50 = 4 nM T31391 C70KAO 44418211 IC50 = 42 nM T31391 C8LC2A 44418213 IC50 = 127 nM T31391 CTM1Y8 44418214 IC50 = 269 nM T31391 C1EMA5 44418215 IC50 = 144 nM T31391 CWDH12 44418216 IC50 = 1300 nM T31391 C1FB4K 44418218 IC50 = 252 nM T31391 CVC3R4 44418219 IC50 = 236 nM T31391 CU1FG2 44418222 IC50 = 247 nM T31391 C8ZH5R 44418223 IC50 = 320 nM T31391 CA9YM3 44418225 IC50 = 232 nM T31391 CQE5Y0 44418229 IC50 = 181 nM T31391 CID62U 44418230 Ki = 4300 nM T31391 CI2H7Q 44418231 Ki = 9080 nM T31391 C2LXS7 44418232 IC50 = 118 nM T31391 CXCV19 44418233 Ki = 7391 nM T31391 CZW38C 44418239 Ki = 9500 nM T31391 C7KF0X 44418240 Ki = 4600 nM T31391 C8QJ7H 44418242 Ki = 19500 nM T31391 C60KPZ 44418243 Ki = 11300 nM T31391 CMKW39 44418246 Ki = 68 nM T31391 CEBQ24 44418249 Ki = 1430 nM T31391 C59HZQ 44418251 IC50 = 8000 nM T31391 CDX2Q5 44418253 Ki = 451000 nM T31391 C0RV8O 44418254 Ki = 182000 nM T31391 C37KEO 44418255 Ki = 6871 nM T31391 C2UR9X 44418256 IC50 = 239 nM T31391 CK20CA 44418257 IC50 = 190 nM T31391 CO3GL6 44418260 IC50 = 207 nM T31391 CY3O7C 44418261 IC50 = 197 nM T31391 C0ITV9 44418262 IC50 = 433 nM T31391 CGR3H7 44418263 IC50 = 21000 nM T31391 C68SHD 44418264 IC50 = 253 nM T31391 CDI98V 44418265 IC50 = 225 nM T31391 CHO5P1 44418266 IC50 = 911 nM T31391 C95XQC 44418268 IC50 = 174 nM T31391 CE3C4D 44420996 Ki = 140 nM T31391 CI2P6M 44420998 Ki = 6.1 nM T31391 C0FT8Q 44420999 Ki = 4 nM T31391 C7VU1I 44421000 Ki = 13 nM T31391 C38PJE 44421001 Ki = 2.3 nM T31391 CX4C3Y 44421002 Ki = 11 nM T31391 CF52AI 44421003 Ki = 23 nM T31391 C6NV0S 44421004 Ki = 1.6 nM T31391 C5W8VX 44421005 Ki = 2.3 nM T31391 C8KC3R 44421006 Ki = 3 nM T31391 C16YHQ 44422417 IC50 = 112 nM T31391 C9IRG5 44422418 IC50 = 11 nM T31391 C7XU0J 44422419 IC50 = 7.9 nM T31391 C58WCU 44422439 IC50 = 19.2 nM T31391 C2F9DG 44422440 IC50 = 51.5 nM T31391 CS63GZ 44422443 IC50 = 5.8 nM T31391 C9M5YC 44422444 IC50 = 7 nM T31391 C0J1UX 44422445 IC50 = 45.4 nM T31391 CKFM17 44422448 IC50 = 6.5 nM T31391 C6C3ZF 44422475 IC50 = 147 nM T31391 C9T1KM 44422476 IC50 = 25.2 nM T31391 CN5G6O 44422477 IC50 = 181 nM T31391 CNQC83 44422485 IC50 = 34 nM T31391 C5NK2E 44422486 IC50 > 300 nM T31391 CZ5UW9 44422487 IC50 = 37.2 nM T31391 C6TZM8 44422496 IC50 > 300 nM T31391 CX5M3Q 44422497 IC50 > 300 nM T31391 C86SXN 44422498 IC50 = 154 nM T31391 C4YP0T 44422507 IC50 = 85.9 nM T31391 C1IW2L 44422508 IC50 > 300 nM T31391 CRWM46 44422509 IC50 > 300 nM T31391 CJK1H2 44422513 IC50 = 9.6 nM T31391 C6C5PM 44422514 IC50 = 7.1 nM T31391 C4KSW0 44422518 IC50 = 9.1 nM T31391 CL40CD 44422519 IC50 = 6.4 nM T31391 CY4K6X 44422522 IC50 = 13.6 nM T31391 CZ8TO9 44422523 IC50 = 13.9 nM T31391 CCFT17 44422525 IC50 = 16.8 nM T31391 C0BXJ2 44422526 IC50 = 17 nM T31391 CGB32F 44422527 IC50 = 228 nM T31391 C1N4RA 44422528 IC50 = 26.4 nM T31391 C1D7ER 44425490 IC50 = 8 nM T31391 CZ2MB8 44426068 IC50 = 6.6 nM T31391 C8PKO5 44426070 IC50 = 139 nM T31391 CW7QD8 44429116 IC50 = 3.5 nM T31391 C1NF6D 44429117 IC50 = 3.4 nM T31391 CG67NO 44429119 IC50 = 5.7 nM T31391 CT54EH 44429120 IC50 = 2.9 nM T31391 C37SUV 44429122 IC50 = 2.4 nM T31391 C57GUJ 44429124 IC50 = 7.8 nM T31391 CW59YC 44429127 IC50 = 3.5 nM T31391 C0L9SG 44429129 IC50 = 6.1 nM T31391 CT2P8M 44429130 IC50 = 9.1 nM T31391 C4KRA5 44429131 IC50 = 3.9 nM T31391 CM2FK3 44429132 IC50 = 2.5 nM T31391 CEL8D9 44429133 IC50 = 3.3 nM T31391 CX48BO 44429134 IC50 = 8.3 nM T31391 CWF04T 44429135 IC50 = 23 nM T31391 CN68CG 44429136 IC50 = 8.9 nM T31391 C6J3CS 44429137 IC50 = 22 nM T31391 C6F1NE 44429138 IC50 = 4.9 nM T31391 CL2G7Z 44429139 IC50 = 7.1 nM T31391 CHT96Z 44429140 IC50 = 5.3 nM T31391 CVD9U0 44429602 IC50 = 3.8 nM T31391 C17MKX 44429603 IC50 = 16 nM T31391 C3SKR2 44429609 IC50 = 4.5 nM T31391 C0SU2X 44429610 IC50 = 2.4 nM T31391 CGQN20 44429612 IC50 = 7.7 nM T31391 CYGD28 44429613 IC50 = 3.5 nM T31391 CZ7LW9 44429614 IC50 = 4.4 nM T31391 CXJD74 44429616 IC50 = 5.7 nM T31391 C6R2IZ 44429619 IC50 = 6 nM T31391 C0A2CF 44429620 IC50 = 4 nM T31391 C4EH0L 44429622 IC50 = 4.9 nM T31391 CY4MF9 44429623 IC50 = 8.3 nM T31391 C02JQU 44429624 IC50 = 11 nM T31391 CG3C7E 44429625 IC50 = 4.3 nM T31391 CHNV25 44429626 IC50 = 4.8 nM T31391 C7IL3S 44431164 IC50 = 98 nM T31391 C0UOS8 44431165 IC50 = 135 nM T31391 CEG05S 44431166 IC50 = 272 nM T31391 CO8S3Z 44431170 IC50 = 805 nM T31391 C2K4RQ 44431176 IC50 = 151 nM T31391 CJZY21 44431177 IC50 = 87 nM T31391 CSJI40 44431185 IC50 = 1018 nM T31391 C36EJR 44431188 IC50 = 486 nM T31391 C2MCA1 44431191 IC50 = 366 nM T31391 C89XVB 44431197 IC50 = 511 nM T31391 CK76EP 44431199 IC50 = 145 nM T31391 C3FPT2 44431200 IC50 = 59 nM T31391 C4F8AG 44431201 IC50 = 264 nM T31391 CWX4I3 44431203 IC50 = 1580 nM T31391 CZ3N9E 44431204 IC50 = 23 nM T31391 C5NAS6 44431205 IC50 = 180 nM T31391 C37SGU 44431206 IC50 = 84 nM T31391 CYD62G 44431212 IC50 = 60 nM T31391 C72WTP 44431213 IC50 = 30 nM T31391 CC3T9G 44431214 IC50 = 65 nM T31391 CL4T3X 44431215 IC50 = 190 nM T31391 C4WVL8 44431216 IC50 = 69 nM T31391 CO08HZ 44431217 IC50 = 37 nM T31391 CCPZ23 44431218 IC50 = 30 nM T31391 C0J7WV 44431219 IC50 = 29 nM T31391 C16ZTV 44431220 IC50 = 219 nM T31391 CR0A1M 44431316 IC50 = 21 nM T31391 CV1R7A 44431317 IC50 = 140 nM T31391 CTB82G 44431744 IC50 = 520 nM T31391 C7O4GL 44431746 IC50 = 35700 nM T31391 CJOR92 44431752 IC50 = 2100 nM T31391 CETI27 44431756 IC50 = 5800 nM T31391 C2VY9T 44431757 IC50 = 142000 nM T31391 C09BFG 44431758 IC50 = 2600 nM T31391 CX3ZH1 44431759 IC50 = 4900 nM T31391 C5JYG0 44431760 IC50 = 26000 nM T31391 C1CRX9 44431761 IC50 = 2300 nM T31391 CB7SA0 44431762 IC50 = 18400 nM T31391 C4FT0P 44431764 IC50 = 8900 nM T31391 C7OJW0 44431765 IC50 = 220 nM T31391 CMU40B 44431766 IC50 = 990 nM T31391 CA9P1R 44431767 IC50 = 1520 nM T31391 CL0VB1 44431768 IC50 = 10590 nM T31391 CHG8I4 44431769 IC50 = 370 nM T31391 C7PLH0 44431770 IC50 = 9380 nM T31391 CC0J6A 44431771 IC50 = 3730 nM T31391 C4X1GA 44431772 IC50 = 5130 nM T31391 C4S8DE 44431773 IC50 = 650 nM T31391 CQX2S0 44431774 IC50 = 32 nM T31391 CL6B7S 44431775 IC50 = 4 nM T31391 C16CRQ 44431776 IC50 = 50 nM T31391 CY76AB 44432858 IC50 = 77 nM T31391 CS95EU 44432859 IC50 = 67 nM T31391 C1PX9V 44432860 IC50 = 223 nM T31391 C3AN4E 44432861 IC50 = 7939 nM T31391 CE4Q5X 44432862 IC50 = 35 nM T31391 CHN6E3 44432863 IC50 = 63 nM T31391 CF2AT6 44432881 IC50 = 15 nM T31391 CTD24F 44432889 IC50 = 95 nM T31391 CSC2E0 44432894 IC50 = 210 nM T31391 CU67PL 44432901 IC50 = 224 nM T31391 C35GZP 44432904 IC50 = 84 nM T31391 C21UQD 44432911 IC50 = 53 nM T31391 CU27DF 44432914 IC50 = 680 nM T31391 C9E1SZ 44432915 IC50 = 339 nM T31391 CZ47KB 44432929 IC50 = 20 nM T31391 CS5BT9 44432935 IC50 = 56 nM T31391 CI9M8R 44432936 IC50 = 17 nM T31391 C5LTR0 44432937 IC50 = 30 nM T31391 C6EJB0 44432938 IC50 = 10 nM T31391 CJ7YN0 44432940 IC50 = 255 nM T31391 CVZ3I2 44432942 IC50 = 47 nM T31391 CT29BC 44432944 IC50 = 25 nM T31391 CNOW68 44433160 IC50 = 140 nM T31391 CJUH82 44433161 IC50 = 2000 nM T31391 C8A1ZL 44433162 IC50 = 150 nM T31391 CJ61CN 44433163 IC50 > 3000 nM T31391 C20OBQ 44433164 IC50 > 3000 nM T31391 C1GBW2 44433165 IC50 > 3000 nM T31391 CEJC97 44433166 IC50 > 3000 nM T31391 CI1NU4 44433167 IC50 = 1000 nM T31391 C5NAI2 44433168 IC50 > 3000 nM T31391 C7TWF9 44433169 IC50 > 3000 nM T31391 C5YUC3 44433174 Ki = 1420 nM T31391 CI5UK4 44433203 IC50 = 790 nM T31391 CVL2Q7 44433204 IC50 = 1400 nM T31391 CR5X3V 44433205 IC50 = 2300 nM T31391 CGB9I5 44433206 IC50 = 2900 nM T31391 CZGM71 44433207 IC50 > 3000 nM T31391 C8PBJ4 44433208 IC50 > 3000 nM T31391 CQ71FG 44433209 IC50 > 3000 nM T31391 C3QOB8 44433210 IC50 > 3000 nM T31391 CO8WI2 44433212 IC50 > 3000 nM T31391 COC75P 44433213 IC50 > 3000 nM T31391 CIB5K2 44433214 IC50 > 3000 nM T31391 C7LI5A 44433215 IC50 > 3000 nM T31391 CCT2I4 44433216 IC50 = 260 nM T31391 CTA59M 44433217 IC50 = 93 nM T31391 CY73TI 44433218 IC50 = 230 nM T31391 C91CFD 44433219 IC50 = 57 nM T31391 CAN07M 44433220 IC50 = 180 nM T31391 C4UTL0 44433221 IC50 = 190 nM T31391 C8CWB2 44433222 IC50 = 37 nM T31391 C4O8SB 44433223 IC50 = 19 nM T31391 CQDS95 44433224 IC50 = 14 nM T31391 CNW1S2 44433225 IC50 = 47 nM T31391 CB04FG 44433226 IC50 = 470 nM T31391 C90GFZ 44433227 IC50 = 130 nM T31391 CSHA84 44433228 IC50 = 160 nM T31391 C6ZP3F 44433229 IC50 = 51 nM T31391 C7KR9C 44433230 IC50 = 120 nM T31391 CH96JN 44433231 IC50 = 71 nM T31391 CR7CQ3 44433232 IC50 = 1300 nM T31391 CWI98S 44433233 IC50 = 32 nM T31391 C23ZRQ 44433234 IC50 = 14 nM T31391 C43RDG 44433235 IC50 = 120 nM T31391 CU6O4S 44433236 IC50 = 70 nM T31391 C8U4QI 44433237 IC50 = 31 nM T31391 C9GIE3 44433617 IC50 = 16 nM T31391 C5B4HS 44433618 IC50 = 12 nM T31391 CU6XZ5 44433646 IC50 = 100 nM T31391 CM8E2D 44433661 IC50 = 38 nM T31391 C07PZD 44433929 Ki > 10000 nM T31391 CG8QR0 44433931 Ki = 3653 nM T31391 CMG6W7 44433932 Ki = 877 nM T31391 CMUR94 44433933 Ki > 10000 nM T31391 CU7AR9 44433934 Ki = 3007 nM T31391 C1ML6S 44433935 Ki > 10000 nM T31391 CM9V3B 44433936 Ki > 10000 nM T31391 C0PLN8 44433937 Ki > 10000 nM T31391 CE5F7Q 44433938 Ki > 10000 nM T31391 CCBR97 44433939 Ki > 10000 nM T31391 CCEO15 44433941 Ki > 10000 nM T31391 CL6V0G 44433942 Ki > 10000 nM T31391 CB70WG 44433943 Ki > 10000 nM T31391 CC02JQ 44433944 Ki > 10000 nM T31391 C9SO3Y 44433945 Ki = 3257 nM T31391 CU7WB6 44433946 Ki > 10000 nM T31391 CAD8G1 44433950 Ki = 1010 nM T31391 C1P2BE 44433951 Ki = 1065 nM T31391 CZA08G 44433952 Ki = 530 nM T31391 CIJF53 44433953 Ki = 731 nM T31391 CTF97G 44433954 Ki = 356 nM T31391 CQ9JD6 44433955 Ki > 10000 nM T31391 CP0M9W 44433956 Ki > 10000 nM T31391 CQ41OU 44433957 Ki = 112 nM T31391 CI15HN 44433958 Ki = 152 nM T31391 C1C9SZ 44433959 Ki = 1944 nM T31391 CA4VY1 44433960 Ki = 3311 nM T31391 CU69GM 44433961 Ki > 10000 nM T31391 CDF80C 44433962 Ki > 10000 nM T31391 CKN0C1 44433969 Ki = 3081 nM T31391 C53UEG 44434115 IC50 = 8 nM T31391 CE92DA 44435310 IC50 = 261000 nM T31391 C3SBK5 44435313 IC50 = 8000 nM T31391 CX7UN0 44435314 IC50 = 4200 nM T31391 CE7XI5 44435315 IC50 > 50000 nM T31391 CGAR49 44435316 IC50 > 250000 nM T31391 C17HRW 44439324 IC50 = 127 nM T31391 C1JQ8Y 44439325 IC50 = 47.6 nM T31391 CAOY46 44439326 IC50 = 13.9 nM T31391 C8XU3A 44439327 IC50 = 57.5 nM T31391 CI7SP9 44439328 IC50 = 10.9 nM T31391 CWG07L 44439329 IC50 = 30.5 nM T31391 CT9V8F 44439330 IC50 = 21 nM T31391 C74ANZ 44439331 IC50 = 13.5 nM T31391 C4B5DI 44439332 IC50 = 12.2 nM T31391 C7LEY1 44439333 IC50 = 8.7 nM T31391 CCJ8T1 44439334 IC50 = 4.1 nM T31391 CWU62R 44439335 IC50 = 10.8 nM T31391 CWG89M 44439336 IC50 = 8.2 nM T31391 CEL4H9 44439337 IC50 = 1.6 nM T31391 C4H3EF 44439338 IC50 = 4.3 nM T31391 C3MLU4 44439339 IC50 = 6.8 nM T31391 C8P1AX 44439340 IC50 = 3 nM T31391 C54TPV 44439341 IC50 = 1.3 nM T31391 CEP51V 44439342 IC50 = 5.6 nM T31391 C4YWH2 44439343 IC50 = 2.3 nM T31391 C1G5PI 44439344 IC50 = 2.4 nM T31391 C02LBF 44439345 IC50 = 2.7 nM T31391 CBE1D5 44439346 IC50 = 3.1 nM T31391 C5T7XF 44439347 IC50 = 2.5 nM T31391 CMC8H4 44439348 IC50 = 1.6 nM T31391 CX4MT0 44439350 IC50 = 1.5 nM T31391 C0OJ1T 44439353 IC50 = 1 nM T31391 C9T6FK 44439354 IC50 = 1.2 nM T31391 C69XIH 44439668 IC50 = 990 nM T31391 CDF76U 44439670 IC50 = 500 nM T31391 C6E8JI 44440627 Ki = 2700 nM T31391 CUQ7K0 44440629 Ki = 280 nM T31391 CSXH19 44440630 Ki = 610 nM T31391 CSI93Z 44440631 Ki = 490 nM T31391 COP6M3 44440633 Ki = 790 nM T31391 C5GKC8 44440634 Ki = 210 nM T31391 CTI8C4 44440635 Ki = 430 nM T31391 C2VAG9 44440645 Ki = 17 nM T31391 CTQR78 44440647 Ki = 20 nM T31391 C08ZST 44440659 Ki = 1 nM T31391 CA9WC3 44440660 Ki = 85 nM T31391 CXC50E 44440661 Ki = 7 nM T31391 CR3PM7 44440662 Ki = 1.7 nM T31391 CB4Q0H 44440663 Ki = 3.4 nM T31391 C6YEQ8 44440664 Ki = 9 nM T31391 CCSI57 44440665 Ki = 1.3 nM T31391 CR4B1M 44443293 IC50 = 30 nM T31391 CY16JP 44443294 IC50 = 38 nM T31391 CN24IJ 44443296 IC50 = 40 nM T31391 C8DSC1 44443297 IC50 = 42 nM T31391 C4F5JW 44443298 IC50 = 47 nM T31391 CJ0G3N 44443299 IC50 = 49 nM T31391 C9F7NQ 44443300 IC50 = 62 nM T31391 C7QCO2 44443301 IC50 = 79 nM T31391 CCQ82F 44443302 IC50 = 86 nM T31391 C1M5TF 44443309 IC50 = 27 nM T31391 CSAE59 44443313 IC50 = 50 nM T31391 CK5E8V 44443319 IC50 = 69 nM T31391 CD0NM4 44443335 IC50 = 78 nM T31391 CEF6H5 44443336 IC50 = 80 nM T31391 CTIM25 44443338 IC50 = 81 nM T31391 CE9Q7A 44443341 IC50 = 83 nM T31391 CI8Q5O 44443343 IC50 = 91 nM T31391 C0MOV3 44443346 IC50 = 2.4 nM T31391 C52VPZ 44443347 IC50 = 3.2 nM T31391 CJ8P7U 44443348 IC50 = 3.3 nM T31391 C8U1XN 44443349 IC50 = 3.6 nM T31391 CM5WU9 44443350 IC50 = 5.3 nM T31391 CB9IM0 44443351 IC50 = 5.4 nM T31391 C8WI4F 44443352 IC50 = 6.2 nM T31391 C3NI8P 44443353 IC50 = 6.7 nM T31391 C7M0HV 44443354 IC50 = 8.5 nM T31391 C0UG4R 44443355 IC50 = 10 nM T31391 C7B5HK 44443356 IC50 = 10 nM T31391 C2G1PX 44443357 IC50 = 3 nM T31391 C3AUF2 44443358 IC50 = 3.4 nM T31391 C0WO5B 44443359 IC50 = 3.5 nM T31391 CUG6X5 44443360 IC50 = 5.5 nM T31391 CARK80 44443361 IC50 = 5.3 nM T31391 CP7WL5 44443363 IC50 = 1.1 nM T31391 C4V0SN 44443364 IC50 = 4.7 nM T31391 CQL53Y 44443365 IC50 = 46 nM T31391 CD2L9G 44443366 IC50 = 3.8 nM T31391 CPN7J9 44443420 IC50 = 65 nM T31391 CI4VR8 44443421 IC50 > 3 nM T31391 CA0NZ7 44443707 IC50 = 140 nM T31391 C24ZHB 44443708 IC50 = 150 nM T31391 C8R4OD 44443709 IC50 = 130 nM T31391 CLDN63 44443710 IC50 = 180 nM T31391 C7LNP2 44443711 IC50 = 230 nM T31391 CJX2M7 44443712 IC50 = 220 nM T31391 C6RST0 44443713 IC50 = 260 nM T31391 C3YL9X 44443714 IC50 = 250 nM T31391 CRH8M1 44443715 IC50 = 250 nM T31391 CIB50E 44443717 IC50 = 130 nM T31391 CK6QF4 44443719 IC50 = 280 nM T31391 CX6O1P 44443720 IC50 = 65 nM T31391 C0YV2D 44443723 IC50 = 610 nM T31391 C1BUJ5 44443725 IC50 = 570 nM T31391 CXS34I 44443727 IC50 = 50 nM T31391 CCHS17 44443729 IC50 = 110 nM T31391 C39KZG 44443736 IC50 = 250 nM T31391 C5H8EJ 44443737 IC50 = 370 nM T31391 CS3Y1G 44444344 IC50 = 100 nM T31391 CL2U9C 44444352 IC50 = 68 nM T31391 C8VE5T 44444353 IC50 = 274 nM T31391 C8F5HC 44444371 IC50 = 4 nM T31391 CEW50M 44444373 IC50 = 4 nM T31391 CO0M7Y 44444375 IC50 = 7 nM T31391 CS93BI 44444377 IC50 = 12 nM T31391 C9J4FB 44444379 IC50 = 14 nM T31391 C3YA4K 44444383 IC50 = 18 nM T31391 C75OIP 44444386 IC50 = 2 nM T31391 C4J6ZG 44444390 IC50 = 4 nM T31391 C05EBU 44444391 IC50 = 2 nM T31391 CSN27E 44445042 IC50 = 5.7 nM T31391 CGN61Q 44445047 IC50 = 1.5 nM T31391 CYW8E3 44445051 IC50 = 2.8 nM T31391 CRG64M 44445053 IC50 = 0.66 nM T31391 C6ZID3 44445055 IC50 = 0.43 nM T31391 C72KOR 44445057 IC50 = 438 nM T31391 C0RTA6 44445060 IC50 = 0.46 nM T31391 CIK8G3 44445063 IC50 = 0.32 nM T31391 CN05VX 44445065 IC50 = 6.3 nM T31391 COA90R 44445067 IC50 = 132 nM T31391 CHRX61 44445075 IC50 > 36900 nM T31391 C6C5IN 44448853 IC50 = 559 nM T31391 CB7MS5 44448857 IC50 = 582 nM T31391 C4IXY7 44448987 IC50 = 2 nM T31391 COP51N 44448988 IC50 = 1 nM T31391 C8KW2A 44448989 IC50 = 99 nM T31391 C9ZRP1 44449015 IC50 = 19 nM T31391 C7E4ZI 44449016 IC50 = 107 nM T31391 CKM5H1 44449017 IC50 = 52 nM T31391 CJ2WY0 44449038 IC50 = 4 nM T31391 C8F2SQ 44449064 IC50 = 2 nM T31391 C7PBF3 44449092 IC50 = 15 nM T31391 CUM32L 44449149 IC50 = 1 nM T31391 CK5M4R 44451509 IC50 = 56 nM T31391 CWI3J9 44451511 IC50 = 41 nM T31391 CEFD93 44451512 IC50 = 600 nM T31391 CKCF72 44451863 IC50 = 51 nM T31391 CR51UD 44451910 IC50 = 60 nM T31391 C76NDG 44451911 IC50 = 16 nM T31391 C20LHD 44452002 IC50 = 13000 nM T31391 CODZ87 44452030 IC50 = 110 nM T31391 CV0Z4T 44452035 IC50 = 70 nM T31391 C7RI2V 44452075 IC50 = 16 nM T31391 CUC93Q 44452076 IC50 = 1100 nM T31391 CK5DW6 44453458 IC50 = 30 nM T31391 C3X8BJ 44453460 IC50 = 42 nM T31391 CDF8R2 44453520 IC50 = 50000 nM T31391 CVO9F2 44453648 IC50 = 57 nM T31391 C91FSI 44453672 IC50 = 90 nM T31391 C5UET4 44453690 IC50 = 645 nM T31391 C2JE8C 44453692 IC50 = 1165 nM T31391 C6EC4J 44453922 IC50 = 12 nM T31391 C4C6NK 44453968 IC50 = 93 nM T31391 CDS52W 44453970 IC50 = 3.2 nM T31391 C9V2HU 44454016 IC50 = 50 nM T31391 CW4H0F 44455959 IC50 = 52 nM T31391 C0S2TV 44455961 IC50 = 21 nM T31391 CH04ND 44455993 IC50 = 37 nM T31391 C50MTS 44456000 IC50 = 604 nM T31391 CQF6O5 44456002 IC50 = 620 nM T31391 CFZB21 44456030 IC50 = 1900 nM T31391 CI0K1D 44456032 IC50 = 340 nM T31391 CYN5Z3 44456147 IC50 = 310 nM T31391 C1WBL5 44456148 IC50 = 350 nM T31391 C3HE5Z 44456310 IC50 = 670 nM T31391 CHKT64 44458509 IC50 = 830 nM T31391 CXWQ16 44458510 IC50 = 360 nM T31391 CBSZ02 44458521 IC50 = 88 nM T31391 CIA6J1 44458523 IC50 = 56 nM T31391 C6LKZ7 44458534 IC50 = 27 nM T31391 CR41OX 44458540 IC50 = 870 nM T31391 CNK09O 44458542 IC50 = 70 nM T31391 CM65HC 44458548 IC50 = 23 nM T31391 CKM0F5 44458549 IC50 = 75 nM T31391 CR4CP3 44458554 IC50 = 21 nM T31391 CU68KW 44458566 IC50 = 270 nM T31391 CC7I6Y 44458573 IC50 = 110 nM T31391 CCI52U 44458574 IC50 = 250 nM T31391 C0K7EZ 44458575 IC50 = 210 nM T31391 CNK64C 44458581 IC50 = 250 nM T31391 CF7I9V 44458586 IC50 = 67 nM T31391 CW7QX0 44458587 IC50 = 55 nM T31391 CJ7Y6A 44458592 IC50 = 35 nM T31391 C9QMB2 44458594 Ki = 56 nM T31391 CPJW14 44458603 Ki = 128 nM T31391 C0K2SV 44458617 Ki = 28 nM T31391 CSIL15 44458629 IC50 = 54 nM T31391 C3EZ1V 44458770 IC50 = 89 nM T31391 COHJ95 44560137 IC50 = 252 nM T31391 CAY0V7 44560138 IC50 = 7.3 nM T31391 C8LNP1 44560139 IC50 = 6.2 nM T31391 CUJR76 44560140 IC50 = 22 nM T31391 C0V4UW 44560141 IC50 = 8.6 nM T31391 CFX7Y2 44560154 IC50 = 12 nM T31391 CGW57E 44560155 IC50 = 88 nM T31391 C0Z5AB 44560156 IC50 = 16 nM T31391 C9JL5Y 44560157 IC50 = 27 nM T31391 C4NC6K 44560158 IC50 = 2.9 nM T31391 CHJ2I3 44560159 IC50 = 7.8 nM T31391 CR4AD0 44560160 IC50 = 8.7 nM T31391 CO9I7S 44560169 IC50 = 13 nM T31391 CD6H2S 44560170 IC50 > 316 nM T31391 C9QC1W 44560171 IC50 = 33 nM T31391 CNF05Y 44560172 IC50 = 3.1 nM T31391 CB73HS 44560173 IC50 = 2.6 nM T31391 CC9B5Y 44560174 IC50 = 3.3 nM T31391 C41LTG 44560184 IC50 = 4.1 nM T31391 C7E1TG 44560185 IC50 = 3.1 nM T31391 C8Z2AR 44560186 IC50 = 3.1 nM T31391 CX3EK8 44560187 IC50 = 8.3 nM T31391 C1BX6I 44560188 IC50 = 5.3 nM T31391 CY78ZH 44560250 IC50 = 2.8 nM T31391 CR69YS 44560251 IC50 = 2.7 nM T31391 C60VSL 44560252 IC50 = 2.4 nM T31391 C70CYA 44560253 IC50 = 8.2 nM T31391 C8CED7 44560254 IC50 = 4.5 nM T31391 CC09EL 44560255 IC50 = 5.4 nM T31391 C5MN2V 44560265 IC50 = 2.9 nM T31391 C75KOL 44560266 IC50 = 5.7 nM T31391 CED9I6 44560267 IC50 = 5.8 nM T31391 C9DLI3 44560268 IC50 = 13 nM T31391 CU65ER 44560279 IC50 = 109 nM T31391 C17LFS 44560280 IC50 = 75 nM T31391 CTD6U0 44560281 IC50 = 31 nM T31391 CB7V0P 44560282 IC50 > 316 nM T31391 CJ4EN1 44560283 IC50 = 39 nM T31391 C91DWY 44560396 IC50 > 100000 nM T31391 CZ9WJ0 44560397 IC50 > 100000 nM T31391 C0FLU7 44560398 IC50 = 80100 nM T31391 CZ43JR 44560454 IC50 > 100000 nM T31391 CY38QP 44560549 IC50 > 100000 nM T31391 C7IL3K 44560550 IC50 > 100000 nM T31391 CF9J7Z 44560551 IC50 > 100000 nM T31391 C1QAI4 44560552 IC50 > 100000 nM T31391 CK25CG 44560553 IC50 > 50000 nM T31391 C4C9NG 44560554 IC50 > 100000 nM T31391 CKIH45 44560555 IC50 > 100000 nM T31391 C2LW3C 44560595 IC50 > 100000 nM T31391 C47WCK 44560596 IC50 > 100000 nM T31391 CL8AE5 44560597 IC50 > 100000 nM T31391 C1YJ8C 44560648 IC50 > 50000 nM T31391 CY6GU1 44560649 IC50 > 62500 nM T31391 C12EYZ 44560650 IC50 = 178000 nM T31391 C7LY9V 44560651 IC50 > 31250 nM T31391 CG5CB2 44560698 IC50 > 250000 nM T31391 CR56BA 44560699 IC50 = 4970 nM T31391 CAK3U5 44560701 IC50 > 100000 nM T31391 C5OW2C 44560747 IC50 > 500000 nM T31391 CM2GN5 44560748 IC50 > 1000000 nM T31391 C5FSB4 44560749 IC50 > 500000 nM T31391 C5WEG1 44560750 IC50 > 250000 nM T31391 CN0KO4 44560770 IC50 = 22 nM T31391 CZSO82 44560823 Ki = 4900 nM T31391 C4IVD9 44560824 IC50 = 37000 nM T31391 C4L3VZ 44560825 IC50 = 15600 nM T31391 CHV7S1 44560826 IC50 = 9700 nM T31391 CE3NF4 44560849 IC50 = 12700 nM T31391 CT6P5E 44560850 IC50 = 16800 nM T31391 CTH9P2 44560851 Ki = 1200 nM T31391 CGZ48C 44560928 IC50 = 51000 nM T31391 C9EK8A 44560929 IC50 > 1000000 nM T31391 CM68VD 44560930 IC50 = 3700 nM T31391 C4SMJ1 44560961 IC50 = 35 nM T31391 C2I3TR 44560962 IC50 = 340 nM T31391 CGV49L 44560963 IC50 = 290 nM T31391 CY0L1G 44560964 IC50 = 2200 nM T31391 C7FST1 44560988 IC50 = 530 nM T31391 CGOM86 44560989 IC50 = 52000 nM T31391 C74ZNK 44560990 IC50 = 2500 nM T31391 C95AUS 44560991 IC50 = 560 nM T31391 CTJ23N 44561008 IC50 = 1300 nM T31391 CR2A0E 44561009 IC50 = 253 nM T31391 C4LQY2 44561010 IC50 = 107 nM T31391 C28XDF 44561011 IC50 = 71 nM T31391 CQ04BE 44561046 IC50 = 9800 nM T31391 C8IF7B 44561117 IC50 = 9200 nM T31391 C29VDX 44561118 IC50 = 200 nM T31391 CB4JA7 44561119 IC50 = 8800 nM T31391 C5K9CX 44561120 IC50 = 55 nM T31391 CQ8DN4 44561152 IC50 = 4400 nM T31391 C4DBU1 44561153 IC50 = 615 nM T31391 C73WBR 44561154 IC50 = 600 nM T31391 CJ91UC 44561155 IC50 = 46 nM T31391 CMO6S2 44561191 IC50 = 20 nM T31391 CF9SB3 44561192 IC50 = 40 nM T31391 C5X1VJ 44561193 IC50 = 120 nM T31391 C31GMV 44561194 IC50 = 85 nM T31391 C1U4YQ 44565237 IC50 = 27 nM T31391 CRK69O 44565238 IC50 = 19 nM T31391 C6M2WD 44565239 IC50 = 21 nM T31391 CTZ9L0 44565254 IC50 = 22 nM T31391 CEMV93 44565274 IC50 = 26 nM T31391 C5E6PQ 44565275 IC50 = 17 nM T31391 CI93OK 44565276 IC50 = 20 nM T31391 C2HRF1 44565277 IC50 = 26 nM T31391 CFEC28 44565466 IC50 = 85 nM T31391 C5MON6 44565467 IC50 = 54 nM T31391 CGA4U6 44565488 IC50 = 64 nM T31391 C1BZ3I 44565489 IC50 = 84 nM T31391 CP3C5F 44565490 IC50 = 75 nM T31391 CRU86T 44565491 IC50 = 62 nM T31391 C3C2DL 44565492 IC50 = 85 nM T31391 CJ2W1P 44565512 IC50 = 60 nM T31391 C5Z9GW 44565513 IC50 = 73 nM T31391 C3I0MO 44565514 IC50 = 86 nM T31391 CI3J6Y 44565535 IC50 = 68 nM T31391 CB90XZ 44565536 IC50 = 101 nM T31391 C01SLH 44565537 IC50 = 24 nM T31391 C8Y2LX 44565538 IC50 = 10 nM T31391 CXD19F 44565539 IC50 = 56 nM T31391 C5BIY6 44565582 IC50 = 309 nM T31391 CFK92H 44565583 IC50 = 25 nM T31391 CE3UT4 44565584 IC50 = 309 nM T31391 CA0O7F 44565585 IC50 = 41 nM T31391 C7LPW8 44565586 IC50 = 134 nM T31391 C39RGP 44565611 IC50 = 338 nM T31391 CPZ7J3 44565844 IC50 = 8.7 nM T31391 C9BGR3 44565845 IC50 = 8.2 nM T31391 CR83QA 44565869 IC50 = 7.4 nM T31391 C6K2WL 44565870 IC50 = 5.6 nM T31391 C3UL2E 44565871 IC50 = 5.2 nM T31391 C9SL5D 44565872 IC50 = 4.8 nM T31391 CZBX95 44565889 IC50 = 31 nM T31391 C1TLY0 44565890 IC50 = 51 nM T31391 CEO20N 44565891 IC50 = 31 nM T31391 COA7X5 44565892 IC50 = 13 nM T31391 CRO3D2 44567651 IC50 = 186 nM T31391 CM95OD 44567652 IC50 = 221 nM T31391 CX6WL5 44567653 IC50 = 27 nM T31391 C4MP9D 44567654 IC50 = 49 nM T31391 CV23FP 44567668 IC50 = 85 nM T31391 CD4C7Y 44567710 IC50 = 123 nM T31391 C4CUJ6 44567711 IC50 = 147 nM T31391 CK1C7W 44567712 IC50 = 78 nM T31391 CTK1I9 44567713 IC50 = 91 nM T31391 C9LQ7N 44567714 IC50 = 1300 nM T31391 CM50CU 44567747 IC50 = 93 nM T31391 C9IF5L 44567748 IC50 > 10000 nM T31391 CMGJ56 44567749 Ki = 5 nM T31391 CR43EI 44567750 Ki = 12 nM T31391 CZ3G4I 44567783 Ki = 31 nM T31391 CNA0I9 44567918 IC50 = 165 nM T31391 C6BXT0 44567919 IC50 = 153 nM T31391 CJ85MG 44567920 IC50 = 110 nM T31391 CUJD19 44567976 IC50 = 38 nM T31391 C5YB6E 44567977 IC50 = 95 nM T31391 CNF09E 44567978 IC50 = 152 nM T31391 C70WEI 44567979 IC50 = 59 nM T31391 CJ0YL5 44568015 IC50 = 2540 nM T31391 CW7NB6 44568016 IC50 = 109 nM T31391 CY8Z3F 44568017 IC50 = 229 nM T31391 CRM76D 44568018 IC50 = 95 nM T31391 C7D4EP 44568055 IC50 = 3430 nM T31391 C3E2UC 44568056 IC50 = 3740 nM T31391 CCG83U 44568057 IC50 = 51 nM T31391 C8XW9A 44568058 IC50 = 31 nM T31391 CMQ7D5 44568097 IC50 = 42 nM T31391 C1F9OL 44568098 IC50 = 63 nM T31391 CUYK75 44568099 IC50 = 92 nM T31391 CZ81XF 44568100 IC50 = 141 nM T31391 C6GT0A 44568134 IC50 = 422 nM T31391 C6IW5D 44568135 IC50 = 630 nM T31391 C3PWD8 44568136 IC50 = 118 nM T31391 C3JBY7 44568137 IC50 = 1715 nM T31391 C4NCA7 44568169 IC50 = 84 nM T31391 C8TXH9 44568170 IC50 = 181 nM T31391 C17PZX 44568171 IC50 = 146 nM T31391 C7SCJ1 44568172 IC50 = 186 nM T31391 CT10GB 44571684 IC50 = 1440 nM T31391 CAT7M0 44571686 IC50 = 510 nM T31391 CSU97M 44571688 IC50 = 3400 nM T31391 C8UGS0 44571690 IC50 = 490 nM T31391 C2WC7S 44571735 IC50 = 410 nM T31391 C0BX2S 44571737 IC50 = 490 nM T31391 C7KYX8 44571739 IC50 = 1392 nM T31391 C2ZYC9 44571741 IC50 = 1500 nM T31391 C68DZI 44571781 IC50 = 350 nM T31391 C1HSU7 44571783 IC50 = 3100 nM T31391 C5WDE4 44571785 IC50 = 405 nM T31391 CB20PW 44571787 IC50 = 387 nM T31391 C8NB2X 44571851 IC50 = 6400 nM T31391 C40YLT 44571853 IC50 = 597 nM T31391 CV9BW0 44571855 IC50 = 423 nM T31391 C0LMD8 44571898 IC50 = 239 nM T31391 CLFG01 44571900 IC50 = 788 nM T31391 C1U5MS 44571902 IC50 = 180 nM T31391 C8DAK4 44571945 IC50 = 288 nM T31391 CM9DP7 44571947 IC50 = 150 nM T31391 CZCU54 44571949 IC50 = 50 nM T31391 CJ96CO 44571951 IC50 = 67 nM T31391 CQW5N2 44571996 IC50 = 260 nM T31391 C7E6IB 44572718 IC50 = 298 nM T31391 CUH81Y 44572719 IC50 = 2 nM T31391 CJHR19 44572720 IC50 = 10 nM T31391 CG71OU 44572782 IC50 = 1600 nM T31391 CG86WR 44580460 IC50 = 13000 nM T31391 C7NP1S 44580497 IC50 = 12000 nM T31391 CQU6S5 44580498 IC50 = 50000 nM T31391 C9JY0C 44580499 IC50 = 180000 nM T31391 CT1N3H 44580500 IC50 = 390000 nM T31391 CYO50L 44580540 IC50 = 11 nM T31391 CSX3I9 44580589 IC50 = 25 nM T31391 CGB0H3 44580664 IC50 = 21 nM T31391 CPR2S7 44589876 IC50 = 7800 nM T31391 C3H0AD 44589877 IC50 = 1000 nM T31391 CY5TC1 44589878 IC50 = 2200 nM T31391 CKM0Z1 44589879 IC50 = 870 nM T31391 CPU4J0 44589931 IC50 = 2500 nM T31391 C4X9GH 44589932 IC50 = 3300 nM T31391 C2DQ0C 44589933 IC50 = 570 nM T31391 C27TUB 44589934 IC50 = 470 nM T31391 CUZ3P0 44589935 IC50 = 190 nM T31391 CM18AD 44589985 IC50 = 64 nM T31391 C4LEZ6 44589986 IC50 = 13 nM T31391 CW2T9J 44589987 IC50 = 12 nM T31391 C1SK7V 44590037 IC50 = 2.7 nM T31391 C6NE1Y 44590038 IC50 = 3.3 nM T31391 CGV2A7 44590039 IC50 = 270 nM T31391 C1KC3N 44590040 IC50 = 35 nM T31391 CZGQ12 44590126 IC50 = 130 nM T31391 CV7RD4 44590127 IC50 = 70 nM T31391 CIE7S0 44590128 IC50 = 350 nM T31391 CCK2S8 44590129 IC50 = 1 nM T31391 C39MKI 44590183 IC50 = 0.64 nM T31391 C82PIC 44590184 IC50 = 1.9 nM T31391 C85SFW 44590185 IC50 = 0.79 nM T31391 C48MPJ 44590596 IC50 = 251 nM T31391 CYE25R 44590598 Ki = 3.6 nM T31391 CI98LA 44590648 IC50 = 22 nM T31391 CBAH06 44590649 IC50 = 6.2 nM T31391 C5R9NI 44590650 IC50 = 0.13 nM T31391 C0W2FC 44590651 IC50 = 0.15 nM T31391 CRN4U5 44590696 IC50 = 4.3 nM T31391 CTC24F 44590734 IC50 = 8 nM T31391 C8CRO4 44590736 IC50 = 18 nM T31391 C91FTW 44591848 IC50 = 18 nM T31391 CY78PR 44591849 IC50 = 22 nM T31391 CE2LW5 44591850 IC50 = 27 nM T31391 CZW0V4 44592369 IC50 > 30000 nM T31391 C3WJ6O 44592370 IC50 = 1930 nM T31391 C07LHO 44592439 IC50 = 3580 nM T31391 CTC4G9 44592440 IC50 > 30000 nM T31391 CIVD36 44592441 IC50 = 25900 nM T31391 C65OXJ 44592442 IC50 > 30000 nM T31391 C8Z0CX 44592443 IC50 = 3250 nM T31391 C9PL5R 44592444 IC50 = 1420 nM T31391 C7L8UN 44592445 IC50 > 30000 nM T31391 CQG62W 44592506 IC50 = 1970 nM T31391 CQHL54 44592507 IC50 = 272 nM T31391 CV42SK 44592508 IC50 = 270 nM T31391 C82YQS 44592509 IC50 = 35 nM T31391 CWJ2U0 44592510 IC50 = 26 nM T31391 CQI40A 44592511 IC50 = 19 nM T31391 CY8R3Q 44593399 IC50 = 115000 nM T31391 CP8YC3 44593408 IC50 = 161000 nM T31391 C4L6NS 44593409 IC50 = 245000 nM T31391 CI0FT1 44593463 IC50 = 47 nM T31391 CAWO01 44593726 IC50 = 6030 nM T31391 CY7Q8W 44629524 IC50 = 22 nM T31391 C65KPR 45101722 IC50 = 6.3 nM T31391 CXYT36 45101723 IC50 = 3 nM T31391 C2RNP7 45102670 IC50 = 16 nM T31391 CQ85WF 45263621 Ki = 6 nM T31391 CGZD98 45265711 IC50 = 103 nM T31391 CW09DZ 45265891 Ki = 3.2 nM T31391 CCO76A 45266134 IC50 = 1700 nM T31391 CU4C5P 45266135 IC50 = 20 nM T31391 CLVM20 45266136 IC50 = 19 nM T31391 CIS3Z8 45267371 IC50 = 92 nM T31391 C8H9GV 45267527 IC50 = 3.2 nM T31391 CP9B0W 45267530 IC50 = 15 nM T31391 C3GJK0 45267531 IC50 = 5.4 nM T31391 CD67HE 45268222 IC50 = 47 nM T31391 CN38QU 45268229 IC50 = 12 nM T31391 CEQ16V 45268233 IC50 = 8 nM T31391 CT93EB 45268323 IC50 = 27 nM T31391 C0QB1V 45268417 IC50 = 2 nM T31391 C2S9ZT 45268436 IC50 = 27 nM T31391 C60MVX 45269112 IC50 = 66 nM T31391 CV7IL1 45269122 IC50 = 24 nM T31391 CX8WC0 45269123 IC50 = 30 nM T31391 C9HR0K 45269274 IC50 = 7.8 nM T31391 CZ1N2O 45269275 IC50 = 12 nM T31391 CIE21V 45269276 IC50 = 5.6 nM T31391 C2W6MT 45269961 IC50 = 87 nM T31391 CWT60M 45269971 IC50 = 14 nM T31391 C4CG2K 45269976 IC50 = 27 nM T31391 CK5P9W 45269994 IC50 = 152 nM T31391 C2A8WO 45269995 IC50 > 16000 nM T31391 C8QJ7X 45270108 IC50 = 7.1 nM T31391 CYWK62 45270115 IC50 = 10 nM T31391 C6E7PR 45270793 IC50 = 92 nM T31391 C6B0CO 45270800 IC50 = 20 nM T31391 CS89DP 45270806 IC50 = 53 nM T31391 CZI9A4 45270821 IC50 > 1600 nM T31391 CQM4X3 45270889 IC50 = 49 nM T31391 CGF7Z6 45270958 IC50 = 2.7 nM T31391 CH5S8Y 45270959 IC50 = 2.2 nM T31391 CM80NZ 45271662 IC50 > 1600 nM T31391 C5NH6Q 45271791 IC50 = 4 nM T31391 C8Z3DK 45271794 IC50 = 3.9 nM T31391 CX62YA 45271796 IC50 = 1.3 nM T31391 CZ8EO2 45271803 IC50 = 3.5 nM T31391 CJ7Q9E 45271813 IC50 = 6.8 nM T31391 CLSJ45 45272523 IC50 = 77 nM T31391 C75XKZ 45272524 IC50 = 27 nM T31391 CSC67Y 45272544 IC50 > 16000 nM T31391 CJI2R6 45272664 IC50 = 2.3 nM T31391 C49BKQ 45272672 IC50 = 5.9 nM T31391 CP36CT 45272682 IC50 = 1.5 nM T31391 C8NL4U 45272683 IC50 = 2.7 nM T31391 CI5AU6 45273390 IC50 = 94 nM T31391 C6S0OC 45273404 IC50 = 8 nM T31391 C2EK3O 45273409 IC50 = 53 nM T31391 C1ZX6U 45273413 IC50 > 1600 nM T31391 CYMR87 45273573 IC50 = 3.5 nM T31391 CFL87A 45273581 IC50 = 6.3 nM T31391 C2XB0P 45273589 IC50 = 6.1 nM T31391 C28PRV 45273594 IC50 = 4.8 nM T31391 CSX2T9 45273602 IC50 = 3.7 nM T31391 CMP59Q 45273603 IC50 = 1.1 nM T31391 C2R3QM 45481268 IC50 = 9 nM T31391 C31XRV 45482320 IC50 = 14130 nM T31391 C28ZXW 45487888 IC50 = 2 nM T31391 C74SVC 45487893 IC50 = 31 nM T31391 C2N3IZ 45487894 IC50 = 3 nM T31391 CP62TC 45487898 IC50 = 4 nM T31391 CPBA81 45487901 IC50 = 90 nM T31391 C0SQW3 45487902 IC50 = 62 nM T31391 CWQ1R9 45487903 IC50 = 2 nM T31391 C8H1KY 45487904 IC50 = 4 nM T31391 C1LJR6 45487907 IC50 = 120 nM T31391 C6X7WJ 45487908 IC50 = 4 nM T31391 CZDS09 45487910 IC50 = 76 nM T31391 CNVU49 45487911 IC50 = 180 nM T31391 C5OXM9 45487915 IC50 = 17 nM T31391 CPJ19X 45487917 IC50 = 2 nM T31391 C16DIR 45487918 IC50 = 28 nM T31391 CV2R7M 45487920 IC50 = 1 nM T31391 C57JRG 45487921 IC50 = 11 nM T31391 C4JD1P 45487922 IC50 = 32 nM T31391 CH30BL 45487925 IC50 = 130 nM T31391 CPB85R 45487926 IC50 = 17 nM T31391 CTY16E 45487930 IC50 = 7 nM T31391 C4QTL9 45487931 IC50 = 5 nM T31391 CG9V0L 45487940 IC50 = 22 nM T31391 C5XTV1 45487945 IC50 = 10 nM T31391 C3VK4G 45487946 IC50 = 2 nM T31391 C0SNL2 46209134 IC50 = 1.6 nM T31391 CE9M5C 46209244 IC50 = 1.6 nM T31391 CW60IG 46209246 IC50 = 1.6 nM T31391 CV65TL 46216691 IC50 = 11 nM T31391 C4QO6X 46216692 IC50 = 0.5 nM T31391 C4GPM1 46229765 IC50 = 61 nM T31391 CCO56J 46229809 IC50 = 38 nM T31391 C0CQM4 46229810 IC50 = 5500 nM T31391 CQ5S8A 46229811 IC50 = 0.5 nM T31391 C6K1YR 46229812 IC50 = 1.7 nM T31391 CU4GE7 46230652 IC50 = 53000 nM T31391 CI4A3C 46230653 IC50 = 19 nM T31391 CEPY06 46231493 IC50 = 1.2 nM T31391 CIEK51 46842529 IC50 = 2810 nM T31391 CDP7Q4 46870369 IC50 = 17 nM T31391 CPH7B4 46871723 IC50 = 8 nM T31391 CDBC45 46890720 IC50 = 180 nM T31391 CLK47C 46890721 IC50 = 23 nM T31391 CS6HL3 46890722 IC50 = 50 nM T31391 C2JY6P 46890723 IC50 = 24 nM T31391 CP7C1L 46890780 IC50 = 26 nM T31391 CED80Z 46890852 IC50 = 93 nM T31391 CA3PE4 46890853 IC50 = 160 nM T31391 CY9T8W 46890854 IC50 = 66 nM T31391 C3TJ0H 46890912 IC50 = 27 nM T31391 CT9HQ6 46890913 IC50 = 24 nM T31391 C9IP7B 46890914 IC50 = 18 nM T31391 CSZE87 46891193 IC50 = 12 nM T31391 C18UES 46891235 IC50 = 59 nM T31391 C23LCY 46891237 IC50 = 65 nM T31391 C57UXS 46891239 IC50 = 80 nM T31391 CIM3K6 46891241 IC50 = 204 nM T31391 C4AUV2 46891291 IC50 = 326 nM T31391 C0UKG7 46891293 IC50 = 121 nM T31391 CJ4G6X 46891342 IC50 = 32 nM T31391 CAL9K6 46891534 IC50 = 15 nM T31391 CPN5T2 46891535 IC50 = 71 nM T31391 C4XTW7 46893990 IC50 > 100000 nM T31391 C8O5VR 46899592 Ki = 8.7 nM T31391 CTY0M5 46899593 Ki = 1 nM T31391 CK9TH1 46899594 Ki = 3.1 nM T31391 C8XD0Q 46899595 Ki = 0.2 nM T31391 CZ84ST 46899596 Ki = 0.5 nM T31391 CPZ70E 46899597 Ki = 0.3 nM T31391 CD3IJ8 46899752 Ki = 0.9 nM T31391 CRK59N 46899753 Ki = 6.6 nM T31391 C6LXU5 46899754 Ki = 2 nM T31391 C52JZL 46899755 Ki = 0.6 nM T31391 C4RC1S 46899756 Ki = 1.8 nM T31391 CP84HR 46899757 Ki = 3.8 nM T31391 CBV4W0 46899937 Ki = 2.6 nM T31391 C5QEJ4 46899938 Ki = 1.1 nM T31391 CHR6V9 46899939 Ki = 2 nM T31391 CQ3A8F 46899940 Ki = 3.2 nM T31391 CX2P8Z 46899941 Ki = 0.7 nM T31391 CC2X1J 46899942 Ki = 2.6 nM T31391 C5QA9M 46900103 Ki = 4 nM T31391 CBI0Q2 46900104 Ki = 0.9 nM T31391 C4IU2E 46900105 Ki = 5 nM T31391 CZEB71 46900106 Ki = 4.7 nM T31391 C2TJW5 46900108 Ki = 1.5 nM T31391 C54ATK 46900259 Ki = 1.3 nM T31391 CI3P6J 46900261 Ki = 2.4 nM T31391 C6DP2G 46900418 Ki = 3.1 nM T31391 CP50DR 46900420 Ki = 5 nM T31391 CF3BL8 46905362 IC50 = 1500 nM T31391 C9JKO5 46905992 IC50 = 21 nM T31391 C8DSG7 46916343 IC50 > 100000 nM T31391 C3RO8F 46916345 IC50 > 100000 nM T31391 CX07LJ 46916346 IC50 > 100000 nM T31391 CF94MW 46916347 IC50 > 100000 nM T31391 CH3F7O 46916384 IC50 > 100000 nM T31391 CM8W6E 46916385 IC50 > 100000 nM T31391 C6FA9Q 46916386 IC50 > 100000 nM T31391 CAW86J 46916387 IC50 > 100000 nM T31391 C63HBE 46916388 IC50 > 100000 nM T31391 CD1CZ7 46916389 IC50 > 100000 nM T31391 CH80LK 46916433 IC50 > 100000 nM T31391 CN4A3P 46916435 IC50 > 100000 nM T31391 CUQ86M 46917047 IC50 > 100000 nM T31391 CS5X9L 46917048 IC50 > 100000 nM T31391 CZP24U 46917049 IC50 = 570 nM T31391 COY5T4 46937042 IC50 = 19 nM T31391 CGMJ52 46938499 IC50 > 100000 nM T31391 C5RAS7 46938602 IC50 > 100000 nM T31391 C3B1LX 46938704 IC50 > 100000 nM T31391 C5TU1F 46938705 IC50 > 100000 nM T31391 CAGP83 46938706 IC50 > 100000 nM T31391 CP9V8Q 46938799 IC50 > 100000 nM T31391 CAB2H9 46938802 IC50 > 100000 nM T31391 C80RAT 47370344 IC50 > 100000 nM T31391 CR5X3K 49785099 IC50 = 0.33 nM T31391 C2HU0V 49785100 IC50 = 1.72 nM T31391 CX7M2K 49785101 IC50 = 0.87 nM T31391 C3XCV4 49785102 IC50 = 1.32 nM T31391 CC8Z5M 49795916 IC50 = 500 nM T31391 CI6U4M 49795917 IC50 = 700 nM T31391 C7HV2K 49795919 IC50 = 2300 nM T31391 CHE51J 49795928 IC50 = 5000 nM T31391 CI6QC3 49795929 IC50 = 800 nM T31391 C8GIY2 49795930 IC50 = 9100000 nM T31391 C2Y5FT 49795931 IC50 = 36 nM T31391 CS1TY7 49795932 IC50 = 23 nM T31391 CUW13V 49795933 IC50 = 47000 nM T31391 CZNL37 49795934 IC50 = 1800000 nM T31391 CGQC72 49795935 IC50 = 31000 nM T31391 CK72BR 49795936 IC50 = 22000 nM T31391 CNB64H 49795937 IC50 = 30 nM T31391 CE2P1Y 49795938 IC50 = 190000 nM T31391 C2TY4D 49795939 IC50 > 10000 nM T31391 COHI43 49795940 IC50 = 400 nM T31391 CDI04P 49795942 IC50 = 1400 nM T31391 CKF3D9 49795943 IC50 = 5000 nM T31391 C95AGZ 49795944 IC50 = 600 nM T31391 CT3XF0 49795948 IC50 = 16 nM T31391 C5RP2S 49796932 IC50 = 510 nM T31391 CZ7A9E 49796933 IC50 = 87 nM T31391 C8D7IG 49796934 IC50 = 539 nM T31391 CBX38D 49796935 IC50 = 1200 nM T31391 CC74RX 49796936 IC50 = 161 nM T31391 CLBU64 49796937 IC50 = 54 nM T31391 C5RF0Y 49796938 IC50 = 7200 nM T31391 CE0C3Y 49796939 IC50 = 75 nM T31391 CI4ZE6 49796940 IC50 = 37 nM T31391 CA54TF 49796941 IC50 = 0.3 nM T31391 CBD8K2 49796942 IC50 = 39 nM T31391 CD21SQ 49796943 IC50 = 170 nM T31391 CODZ18 49796944 IC50 = 118 nM T31391 CI25XP 49796945 IC50 = 721 nM T31391 CF65YQ 49796946 IC50 = 1640 nM T31391 C32MAO 49796947 IC50 = 10 nM T31391 CHJ76U 49796948 IC50 = 3.7 nM T31391 CU25OB 49796949 IC50 = 5.1 nM T31391 C1ZJS7 49796950 IC50 = 4200 nM T31391 C8GWI5 49796951 IC50 = 1.8 nM T31391 CH2W5L 49796952 IC50 = 18 nM T31391 C8WYA5 49796953 IC50 = 0.48 nM T31391 C0P6JR 49796954 IC50 = 1.6 nM T31391 CQH86V 49796955 IC50 = 8.2 nM T31391 C08NMS 49796956 IC50 = 0.83 nM T31391 CR63MS 49796957 IC50 = 18 nM T31391 CJ5FR6 49796958 IC50 = 7.1 nM T31391 C7IBX0 49796959 IC50 = 3300 nM T31391 CU83MS 49796960 IC50 = 12 nM T31391 CQ5YV7 49796961 IC50 = 13 nM T31391 C1T9ON 49796962 IC50 = 3600 nM T31391 C1ZVH6 49796963 IC50 = 82 nM T31391 CB26OQ 49796964 IC50 = 1200 nM T31391 C0NO8F 49796965 IC50 = 9.5 nM T31391 C69JQC 49796966 IC50 = 33 nM T31391 C01RDX 49796967 IC50 = 1.7 nM T31391 C2SXO4 49796968 IC50 = 1.6 nM T31391 C7SH5C 49796969 IC50 = 12 nM T31391 C7K3HC 49796970 IC50 = 295 nM T31391 CBMV50 49796972 IC50 = 64 nM T31391 C8IL0K 49796973 IC50 = 980 nM T31391 CA90LB 49796974 IC50 = 1600 nM T31391 C07DHG 49796977 IC50 = 3500 nM T31391 CAS2P4 49796982 IC50 = 220 nM T31391 CG79KT 49796985 IC50 = 390 nM T31391 C4D8RE 49796990 IC50 = 6.6 nM T31391 CUKB68 49796994 IC50 = 550 nM T31391 CUR9B0 49796995 IC50 = 9.2 nM T31391 CWHO58 49796998 IC50 = 45 nM T31391 CX74RG 49796999 IC50 = 12 nM T31391 C20MAQ 49797000 IC50 = 13 nM T31391 CD67OX 49797001 IC50 = 192 nM T31391 C9LEF5 49797002 IC50 = 9.1 nM T31391 CO2AX9 49797003 IC50 = 3.3 nM T31391 CEM61W 49797006 IC50 = 520 nM T31391 C7Y0JL 49797007 IC50 = 59 nM T31391 CW45IK 49797008 IC50 = 37 nM T31391 C79JUI 49797011 IC50 = 67 nM T31391 CVAK94 49797012 IC50 = 29 nM T31391 CUK5J1 49797013 IC50 = 43 nM T31391 C4ZK5C 49797014 IC50 = 2.2 nM T31391 C1PV8J 49797015 IC50 = 30 nM T31391 C9YEU6 49797016 IC50 = 17 nM T31391 CZD4S2 49797017 IC50 = 99 nM T31391 CKY80F 49797018 IC50 = 11 nM T31391 CS0D8Q 49797021 IC50 = 27 nM T31391 C3GF4M 49797022 IC50 = 100 nM T31391 C8XZT9 49797023 IC50 = 71 nM T31391 C5H2AS 49797024 IC50 = 94 nM T31391 C4P0VW 49797025 IC50 = 20 nM T31391 CVY8M1 49797028 IC50 = 110 nM T31391 CM59HB 49797029 IC50 = 230 nM T31391 CH7Y1J 49797030 IC50 = 44 nM T31391 CX18HI 49797031 IC50 = 21 nM T31391 CUM28Z 49797035 IC50 = 110 nM T31391 COS23G 49797036 IC50 = 7.5 nM T31391 C2TSG6 49797038 IC50 = 56 nM T31391 C7BI3W 49797039 IC50 = 21 nM T31391 C71THK 49797040 IC50 = 1100 nM T31391 C0SG5O 49797041 IC50 = 7900 nM T31391 CM37VB 49797042 IC50 = 170 nM T31391 C51NUG 49797043 IC50 = 480 nM T31391 C65WXC 49797044 IC50 = 600 nM T31391 CHTO37 49797045 IC50 = 2000 nM T31391 CA8R5K 49797046 IC50 = 3700 nM T31391 CLAR35 49797047 IC50 = 250 nM T31391 C9OCZ3 49797048 IC50 = 54000 nM T31391 C49RUW 49797049 IC50 = 1100 nM T31391 C4EHT7 49797050 IC50 = 3700 nM T31391 CW6G5R 49797051 IC50 = 2800 nM T31391 CUK6G0 49797052 IC50 = 120 nM T31391 CJ1FE2 49797053 IC50 = 280 nM T31391 CKJO08 49797054 IC50 = 4200 nM T31391 C70KVU 49797055 IC50 = 3600 nM T31391 CP59BI 49797056 IC50 = 360 nM T31391 CEDL61 49797057 IC50 = 770 nM T31391 C5J2LV 49797058 IC50 = 1400 nM T31391 CEI20Q 49797059 IC50 = 1100 nM T31391 C7B5DY 49797060 IC50 = 6 nM T31391 C5B1RM 49797061 IC50 = 100 nM T31391 C40HJC 49797062 IC50 = 240 nM T31391 CL3P4H 49797063 IC50 = 98 nM T31391 CPC76U 49797064 IC50 = 140 nM T31391 C5F4JN 49797065 IC50 = 580 nM T31391 C86HND 49797066 IC50 = 130 nM T31391 C8E4XD 49797067 IC50 = 1500 nM T31391 CHO1U0 49797068 IC50 = 100 nM T31391 CO1TW7 49797069 IC50 = 69 nM T31391 CAD6W1 49797071 IC50 = 110 nM T31391 CQYU80 49797072 IC50 = 110 nM T31391 CEZ38H 49797073 IC50 = 110 nM T31391 C0CEU7 49797074 IC50 = 140 nM T31391 C72JXY 49797075 IC50 = 27 nM T31391 COA41Q 49797076 IC50 = 510 nM T31391 CPQ3Z2 49797077 IC50 = 140 nM T31391 C1WI0D 49797078 IC50 = 60 nM T31391 C4D8XP 49797079 IC50 = 390 nM T31391 CQG4J6 49797080 IC50 = 130 nM T31391 CKM9S4 49797081 IC50 = 75 nM T31391 C3JRW0 49797082 IC50 = 370 nM T31391 C27IEB 49797083 IC50 = 150 nM T31391 C0JUL3 49797084 IC50 = 110 nM T31391 C85DOL 49797085 IC50 = 110 nM T31391 CEGO30 49797086 IC50 = 150 nM T31391 C2TC3I 49797087 IC50 = 440 nM T31391 C04JWY 49797088 IC50 = 240 nM T31391 CA2U4Y 49797089 IC50 = 56 nM T31391 CFT46J 49797090 IC50 = 37 nM T31391 C35TFW 49797091 IC50 = 86 nM T31391 CRL7Z5 49797092 IC50 = 710 nM T31391 CYU74X 49797093 IC50 = 420 nM T31391 C2O3SG 49797094 IC50 = 150 nM T31391 CFL3O2 49797106 IC50 = 48 nM T31391 CF4NR7 49797107 IC50 = 26 nM T31391 CV9QW6 49797108 IC50 = 31 nM T31391 CJZA65 49797109 IC50 = 1100 nM T31391 CBS36X 49797110 IC50 = 38 nM T31391 C0STP5 49797111 IC50 = 29 nM T31391 C7KV5R 49797112 IC50 = 320 nM T31391 CJPX53 49797113 IC50 = 570 nM T31391 C2OI0Y 49797114 IC50 = 25 nM T31391 CW20FJ 49797115 IC50 = 34 nM T31391 C9P6VU 49797116 IC50 = 49 nM T31391 C67SIA 49797117 IC50 = 74 nM T31391 CCI8Y0 49797118 IC50 = 67 nM T31391 CE10UF 49797119 IC50 = 37 nM T31391 CLH0V3 49797120 IC50 = 120 nM T31391 C2N8WX 49797121 IC50 = 26 nM T31391 CNCE06 49797122 IC50 = 90 nM T31391 C76UAB 49797123 IC50 = 69 nM T31391 CHWT89 49797124 IC50 = 92 nM T31391 C1Z6NE 49797125 IC50 = 61 nM T31391 C25MQG 49797126 IC50 = 229 nM T31391 COL54B 49797127 IC50 = 117 nM T31391 C5OUQ3 49797128 IC50 = 52 nM T31391 C3NMI8 49797173 Ki = 12 nM T31391 C1E3YB 49797174 Ki = 6 nM T31391 CVD0I1 49797175 Ki = 3.6 nM T31391 CH02OC 49797176 Ki = 4.7 nM T31391 CY1OJ5 49797177 Ki = 1.3 nM T31391 CL8TW4 49797178 Ki < 140 nM T31391 C25ZSD 49797191 IC50 = 203 nM T31391 C0OJX9 49797192 IC50 = 8 nM T31391 C7GZ4B 49797193 IC50 = 19 nM T31391 CVT2E5 49797194 IC50 = 40 nM T31391 C75MGE 49797195 IC50 = 13 nM T31391 CVS70C 49797196 IC50 = 13 nM T31391 C42QPW 49797197 IC50 = 70 nM T31391 C6ZGL5 49797198 IC50 = 52 nM T31391 C1B5NH 49797199 IC50 = 31 nM T31391 CGQN24 49797200 IC50 = 560 nM T31391 CS2AI5 49797201 IC50 = 1210 nM T31391 CM7RE3 49797202 IC50 = 1830 nM T31391 CGM9E7 49797203 IC50 = 3050 nM T31391 COU0I6 49797204 IC50 = 19 nM T31391 C3XML2 49797205 IC50 = 19 nM T31391 CP0O2F 49797223 IC50 = 210 nM T31391 CTH7I8 49797224 IC50 = 58 nM T31391 CG9P7O 49797225 IC50 = 144 nM T31391 C3A2QK 49797226 IC50 = 125 nM T31391 C4NOK2 49797227 IC50 = 111 nM T31391 CB13PO 49797228 IC50 = 67 nM T31391 C47VOG 49797229 IC50 = 463 nM T31391 CD2CL1 49797230 IC50 = 650 nM T31391 C0LK6B 49797231 IC50 = 14 nM T31391 CON0A6 49797232 IC50 = 37 nM T31391 C4AVU3 49797233 IC50 = 90 nM T31391 CQ93MI 49797234 IC50 = 82 nM T31391 CO2JV8 49797235 IC50 = 63 nM T31391 C27LDC 49797236 IC50 = 54 nM T31391 CA5GM6 49797237 IC50 = 3700 nM T31391 CT8PW1 49797238 IC50 = 7 nM T31391 CJQ38S 49797239 IC50 = 12 nM T31391 CT65MR 49797240 IC50 = 130 nM T31391 C08IFZ 49797241 IC50 = 43 nM T31391 CA4E8M 49797242 IC50 = 13 nM T31391 CN8FR2 49797243 IC50 = 22 nM T31391 C37MDP 49797244 IC50 = 5 nM T31391 CM41RN 49797245 IC50 = 2 nM T31391 C59JEK 49797246 IC50 = 8 nM T31391 CUMH43 49797248 IC50 = 8 nM T31391 CM59PE 49797249 IC50 = 5 nM T31391 CN5K1S 49797250 IC50 = 31 nM T31391 CT5HY0 49797251 IC50 = 6 nM T31391 C0E5PY 49797252 IC50 = 9 nM T31391 C3E5JB 49797253 IC50 = 16 nM T31391 CA8P5N 49797344 IC50 = 870 nM T31391 CJL2B8 49797345 IC50 = 430 nM T31391 CT79YI 49797346 IC50 = 25 nM T31391 C93VJO 49797347 IC50 = 160 nM T31391 CDI52A 49797348 IC50 = 300 nM T31391 C7ATK9 49797349 IC50 = 160 nM T31391 C2Y3DS 49797350 IC50 = 600 nM T31391 CA4CE3 49797351 IC50 = 150 nM T31391 C3A8YT 49797352 IC50 = 210 nM T31391 C1Z8HB 49797353 IC50 = 48 nM T31391 CC0T8H 49797354 IC50 = 330 nM T31391 C92QND 49797355 IC50 = 1490 nM T31391 C2HPE8 49797356 IC50 = 1280 nM T31391 C9UXH2 49797357 IC50 = 440 nM T31391 CTYO37 49797358 IC50 = 24 nM T31391 C1K4FR 49797359 IC50 = 22 nM T31391 CJ2D0P 49797360 IC50 = 74 nM T31391 CA3Q2W 49797361 IC50 = 29 nM T31391 CNMF62 49797362 IC50 = 21 nM T31391 C3HU6X 49797446 IC50 = 1490 nM T31391 C3U1KQ 49797450 IC50 = 525 nM T31391 C76KMB 49797451 IC50 = 17 nM T31391 C02MPV 49797452 IC50 = 122 nM T31391 CLVF17 49797501 IC50 = 9 nM T31391 CR0AK2 49797502 IC50 = 6 nM T31391 CM1Y7K 49797503 IC50 = 7 nM T31391 CUSI73 49797504 IC50 = 10 nM T31391 CJ0DX6 49797505 IC50 = 22 nM T31391 C2A7LE 49797506 IC50 = 7 nM T31391 CU4M3T 49797507 IC50 = 15 nM T31391 C8GCS5 49797508 IC50 = 17 nM T31391 CTP9L2 49797509 IC50 = 31 nM T31391 CT76PM 49797510 IC50 = 8 nM T31391 C4K0QT 49797511 IC50 = 19 nM T31391 CLHB50 49797512 IC50 = 37 nM T31391 CC56FE 49797513 IC50 = 11 nM T31391 C4T6AB 49797514 IC50 = 8 nM T31391 C41VHF 49797515 IC50 = 31 nM T31391 CBD9H2 49797516 IC50 = 12 nM T31391 CAOC90 49797517 IC50 = 31 nM T31391 C0F5QX 49797518 IC50 = 12 nM T31391 C7T5XW 49797519 IC50 = 16 nM T31391 CM6SF5 49797520 IC50 = 25 nM T31391 CQZN45 49797521 IC50 = 14 nM T31391 CG64BU 49797522 IC50 = 13 nM T31391 C5G3MA 49797524 IC50 = 5 nM T31391 CO42DE 49797525 IC50 = 35 nM T31391 C5L1EP 49797526 IC50 = 40 nM T31391 CTWR80 49797527 IC50 = 6 nM T31391 CPIC42 49797528 IC50 = 7 nM T31391 C5N1ZB 49797529 IC50 = 5 nM T31391 CU72EZ 49797596 IC50 = 17 nM T31391 C6AZ2C 49797599 IC50 = 52 nM T31391 CR86PO 49797604 IC50 = 22 nM T31391 C6DJX7 49797605 IC50 = 4.2 nM T31391 CK3ZI1 49797607 IC50 = 7.1 nM T31391 C7AD0C 49797610 IC50 = 53 nM T31391 C4XHO5 49797612 IC50 = 8 nM T31391 C7VL5U 49797614 IC50 = 28 nM T31391 CY09JE 49797615 IC50 = 47 nM T31391 C1ZLF0 49797616 IC50 = 13 nM T31391 CN48OE 49797627 IC50 = 77 nM T31391 CV6I0O 49797630 IC50 = 14 nM T31391 CAG1U7 49797631 IC50 = 56 nM T31391 C8JNU1 49797636 IC50 = 68 nM T31391 C0DN5G 49797642 IC50 = 47 nM T31391 CJVS96 49797644 IC50 = 18 nM T31391 CBRT78 49797650 IC50 = 8.6 nM T31391 CZW93Y 49797653 IC50 = 30 nM T31391 COM5Q7 49836030 IC50 = 27 nM T31391 CKZJ30 49837952 IC50 = 16 nM T31391 CXR05H 49837954 IC50 = 11 nM T31391 C4QSP1 49837961 IC50 = 10 nM T31391 C1WSF0 49843627 IC50 = 300 nM T31391 C31PHS 49843629 IC50 = 101 nM T31391 CDAK59 49843631 IC50 = 124 nM T31391 CSWR53 49845007 IC50 = 2300 nM T31391 C02RWO 49845009 IC50 = 1060 nM T31391 CG5O9N 49845011 IC50 = 1240 nM T31391 C9ST1E 49845161 IC50 = 460 nM T31391 C64NVQ 49845166 IC50 = 1236 nM T31391 C3CVF2 49845349 IC50 = 360 nM T31391 CTDR85 49862539 Ki = 73 nM T31391 CT8Q9N 49862713 Ki = 73 nM T31391 C0OB8C 49862714 Ki = 50 nM T31391 CJ58AG 49862715 Ki = 50 nM T31391 C42TSR 49862716 Ki = 31 nM T31391 CPU7F6 49862790 Ki = 29 nM T31391 C4FZY2 49862791 Ki = 442 nM T31391 CF40YM 49862792 Ki = 106 nM T31391 CK0GC5 49864113 Ki = 5.4 nM T31391 CK1CD3 50925423 IC50 = 23 nM T31391 C8XA7H 50942035 IC50 = 13 nM T31391 CFT4L5 50970490 IC50 = 93 nM T31391 C7T6PI 50994092 IC50 = 1.1 nM T31391 C67CTP 51032641 IC50 = 88.82 nM T31391 C1ECS9 51050448 IC50 = 66 nM T31391 CL4S9Y 51050450 IC50 = 39 nM T31391 CWZ76P 51050544 IC50 = 23 nM T31391 CT3D7J 51050546 IC50 = 8.7 nM T31391 C5O1PJ 51050548 IC50 = 9.6 nM T31391 CR6ZG8 51050550 IC50 = 6.6 nM T31391 CY3W8O 51051127 IC50 = 57 nM T31391 C2GNK6 51051129 IC50 = 58 nM T31391 CLU39H 51051131 IC50 = 18 nM T31391 C5PRF8 51051132 IC50 = 18 nM T31391 CYF04M 51051134 IC50 = 5.7 nM T31391 CPCY75 51051136 IC50 = 4.4 nM T31391 C7JM3I 51051236 IC50 = 19 nM T31391 CZ5HJ0 51051238 IC50 = 4.6 nM T31391 C1OUG5 51051240 IC50 = 2.5 nM T31391 C6GAP9 51051329 IC50 = 20 nM T31391 C9KPJ6 51051331 IC50 = 10 nM T31391 C85CEJ 51346970 IC50 = 55 nM T31391 C4PFT3 51346971 IC50 = 94 nM T31391 CLG9I5 51355035 IC50 = 89.5 nM T31391 CLND76 51356956 IC50 = 44 nM T31391 CH92AI 51356957 IC50 = 80 nM T31391 CH89VX 51356958 IC50 = 686 nM T31391 C5D4HV 51356959 IC50 = 674 nM T31391 C03ROM 51356960 IC50 < 50000 nM T31391 C8WOG2 51356962 IC50 = 674 nM T31391 CJ0Q4A 52918281 IC50 = 50.66 nM T31391 C4VC2U 52942435 IC50 = 87 nM T31391 C2B6EX 52943488 Ki = 11 nM T31391 CGOM96 52943515 IC50 = 114 nM T31391 C56CXU 52943631 IC50 = 151 nM T31391 CHD7O6 52943758 IC50 = 13 nM T31391 C4I6ML 52944843 IC50 = 23 nM T31391 C57XSM 52944845 IC50 = 122 nM T31391 CT6SQ3 52944941 IC50 = 28 nM T31391 C7RJM9 52945660 IC50 = 10 nM T31391 C9OAF1 52946149 IC50 = 1.8 nM T31391 CBVC96 52946447 IC50 = 10 nM T31391 CC56BV 52946866 IC50 > 100000 nM T31391 CC7N8S 52948914 IC50 = 36 nM T31391 C4LVO6 52948971 IC50 = 12 nM T31391 CTU0J1 52949742 IC50 = 103 nM T31391 CD4HQ1 53233695 IC50 = 3100 nM T31391 C89KWN 53233798 IC50 = 4000 nM T31391 CEFX05 53311069 IC50 = 1100 nM T31391 CQL50R 53311070 IC50 > 100000 nM T31391 C1Q4WK 53311071 IC50 = 20000 nM T31391 C67LHZ 53311072 IC50 = 530 nM T31391 CQ0ZJ2 53311073 IC50 = 5200 nM T31391 C7PMY1 53311074 IC50 = 38000 nM T31391 CWN9H7 53311140 IC50 = 100 nM T31391 CAL51C 53311141 IC50 = 16000 nM T31391 C2SXV0 53311142 IC50 = 88000 nM T31391 C7AEF8 53311143 IC50 > 100000 nM T31391 C5IOZ6 53311144 IC50 = 3400 nM T31391 CVR4H3 53311222 IC50 = 430 nM T31391 CNX08H 53311223 IC50 = 110 nM T31391 CET6W5 53311225 IC50 = 2500 nM T31391 C3RZS4 53311226 IC50 = 480 nM T31391 CHR17Y 53311227 IC50 = 13 nM T31391 C3HGW8 53312238 IC50 > 100000 nM T31391 CM03UX 53312239 IC50 > 100000 nM T31391 C9K4CZ 53312243 IC50 > 100000 nM T31391 CU4BS2 53312323 IC50 = 23000 nM T31391 CF5I6O 53312326 IC50 = 22 nM T31391 C6PSL2 53312327 IC50 > 100000 nM T31391 C0WYS5 53312328 IC50 = 45 nM T31391 CI0Z2A 53317343 IC50 > 50000 nM T31391 CLZ1M4 53317345 IC50 > 50000 nM T31391 CO3SY5 53317346 IC50 > 50000 nM T31391 C4M7TX 53317347 IC50 > 50000 nM T31391 C37HQG 53317348 IC50 > 50000 nM T31391 CYC69Q 53317564 IC50 = 85 nM T31391 C0QOV9 53317565 IC50 = 180 nM T31391 CURC70 53317566 IC50 = 400 nM T31391 C3ZK1W 53317575 IC50 = 120 nM T31391 CBQ0J7 53317579 IC50 = 280 nM T31391 CIY9F7 53317580 IC50 = 57 nM T31391 C5DMS9 53317581 IC50 = 450 nM T31391 C1XD9W 53317582 IC50 = 82 nM T31391 CR0O8T 53317583 IC50 = 18 nM T31391 CHW98L 53317619 IC50 = 13 nM T31391 C9AB1E 53317627 IC50 = 488 nM T31391 C0XQ2B 53318462 IC50 = 22.53 nM T31391 CJO28A 53318492 IC50 = 29.92 nM T31391 C45YDV 53318494 IC50 = 52.34 nM T31391 C6H4ZL 53318496 IC50 = 30.03 nM T31391 CYBP96 53318498 IC50 = 36.43 nM T31391 C9GLH7 53318841 IC50 = 84 nM T31391 C06TDE 53318842 IC50 = 150 nM T31391 C73TER 53318856 IC50 = 110 nM T31391 CC56NE 53318863 IC50 = 110 nM T31391 C4UJI8 53318864 IC50 = 310 nM T31391 C8CZ2A 53318865 IC50 = 110 nM T31391 CLVY47 53318866 IC50 = 51 nM T31391 CQC8N4 53318918 IC50 = 80 nM T31391 C7P2UE 53318921 IC50 = 1400 nM T31391 CP67YM 53318983 IC50 > 50000 nM T31391 C6SJ4Z 53318987 IC50 = 74 nM T31391 CM7S5W 53319067 IC50 = 110 nM T31391 C85NSB 53319824 IC50 = 37.54 nM T31391 CTW2R8 53319826 IC50 = 46.89 nM T31391 CW83TR 53319828 IC50 = 15.8 nM T31391 CC59LI 53319949 IC50 > 50000 nM T31391 CNW4K5 53319950 IC50 > 50000 nM T31391 CQK53D 53319951 IC50 > 50000 nM T31391 CD9LA8 53320113 IC50 > 50000 nM T31391 C1X3NE 53320178 IC50 = 120 nM T31391 C1P8BK 53320179 IC50 = 110 nM T31391 C50UBZ 53320180 IC50 = 140 nM T31391 C2JTR7 53320181 IC50 = 260 nM T31391 C0TYJ5 53320182 IC50 = 77 nM T31391 C7RSX2 53320183 IC50 = 72 nM T31391 CJU34O 53320232 IC50 = 19 nM T31391 C8ML9Y 53321113 IC50 = 45.2 nM T31391 CF0B3T 53321115 IC50 = 46.61 nM T31391 CEO6M2 53321117 IC50 = 22.76 nM T31391 CFPY75 53321119 IC50 = 17.83 nM T31391 CXZ47P 53321201 IC50 < 50000 nM T31391 CJ2V8E 53321202 IC50 = 937 nM T31391 CGVE79 53321203 IC50 < 50000 nM T31391 CP12HY 53321204 IC50 < 50000 nM T31391 C0XLS2 53321252 IC50 < 50000 nM T31391 CNT89R 53321253 IC50 > 50000 nM T31391 CO58YD 53321254 IC50 > 50000 nM T31391 C9XGE4 53321472 IC50 = 140 nM T31391 CY0ZV9 53321485 IC50 = 170 nM T31391 CK0OB2 53321486 IC50 = 38 nM T31391 CNK34J 53321487 IC50 = 260 nM T31391 C7EO3D 53321495 IC50 = 140 nM T31391 C3M7PQ 53321496 IC50 = 850 nM T31391 C0NUQ7 53321497 IC50 = 330 nM T31391 C31DSJ 53321498 IC50 = 450 nM T31391 C2ZKV9 53321499 IC50 = 71 nM T31391 CGA05O 53321545 IC50 = 216 nM T31391 CAU2F0 53321549 IC50 = 12 nM T31391 CB76JK 53321550 IC50 = 59 nM T31391 C50RJL 53321566 IC50 = 13 nM T31391 C3QT0R 53321621 IC50 = 140 nM T31391 CF2GQ1 53321670 IC50 = 22 nM T31391 C4UA2C 53322441 IC50 = 12.4 nM T31391 CF5M0P 53322443 IC50 = 33.17 nM T31391 CQK38R 53322445 IC50 = 33.25 nM T31391 C3OTG6 53322447 IC50 = 47.27 nM T31391 CKT3E2 53322456 IC50 = 77.06 nM T31391 CR9TY2 53322529 IC50 > 50000 nM T31391 C56URQ 53322530 IC50 < 50000 nM T31391 C1ZIS9 53322575 IC50 > 50000 nM T31391 C2MA6T 53322742 IC50 > 50000 nM T31391 CXIS21 53322758 IC50 = 730 nM T31391 CY71QL 53322814 IC50 = 130 nM T31391 CLU96Y 53322820 IC50 = 270 nM T31391 C8YVF1 53322821 IC50 = 290 nM T31391 C4QS6V 53322822 IC50 = 220 nM T31391 C62JTB 53322823 IC50 = 710 nM T31391 CT14FU 53322824 IC50 = 690 nM T31391 CXJ1F8 53322825 IC50 = 670 nM T31391 C3K1VY 53322826 IC50 = 21 nM T31391 CC09IP 53322885 IC50 = 41 nM T31391 C9N6HK 53322952 IC50 = 70 nM T31391 C7NUF3 53323807 IC50 = 28.6 nM T31391 C3QGT8 53323865 IC50 < 50000 nM T31391 C0FOV2 53323866 IC50 < 50000 nM T31391 CZ4I5J 53323915 IC50 < 50000 nM T31391 C4E8OK 53323916 IC50 > 50000 nM T31391 CB7HG9 53323917 IC50 > 50000 nM T31391 C9LU8M 53324129 IC50 = 99 nM T31391 CCY7M0 53324130 IC50 = 130 nM T31391 C4F1QK 53324142 IC50 = 500 nM T31391 CZN71C 53324143 IC50 = 670 nM T31391 CG83JZ 53324144 IC50 = 140 nM T31391 CE8J1D 53324145 IC50 = 140 nM T31391 C0Y3AC 53324153 IC50 = 120 nM T31391 C9O1IW 53324154 IC50 = 910 nM T31391 CTW5G0 53324155 IC50 = 130 nM T31391 C2DPZ0 53324156 IC50 = 54 nM T31391 C9A4JG 53324203 IC50 = 28 nM T31391 CPCE78 53324209 IC50 = 47 nM T31391 C6CJ0H 53324210 IC50 = 1.6 nM T31391 CL5Z8N 53324211 IC50 = 39 nM T31391 CV7UM8 53324212 IC50 = 37 nM T31391 C98EJV 53324213 IC50 = 13 nM T31391 CSN28M 53324293 IC50 = 2400 nM T31391 C2FRA0 53324311 IC50 > 50000 nM T31391 CDW31Y 53325018 IC50 < 50000 nM T31391 C76TDZ 53325194 IC50 < 50000 nM T31391 CJWL87 53325195 IC50 > 50000 nM T31391 CBT0Z8 53325196 IC50 > 50000 nM T31391 C2N5BX 53325197 IC50 > 50000 nM T31391 CF65NE 53325325 IC50 = 77 nM T31391 C25OJW 53325399 IC50 = 430 nM T31391 CXW5O9 53325446 IC50 = 280 nM T31391 C1SO0C 53325447 IC50 = 570 nM T31391 C1S3WB 53325453 IC50 = 200 nM T31391 C2KFW6 53325454 IC50 = 75 nM T31391 C4ZFR5 53325455 IC50 = 78 nM T31391 CPS51R 53325503 IC50 = 153 nM T31391 CW8TM9 53325504 IC50 = 26 nM T31391 CCOQ72 53325553 IC50 = 26.17 nM T31391 C5UB1G 53325568 IC50 < 50000 nM T31391 C1Z4RT 53326344 IC50 = 15.09 nM T31391 CX6Q3E 53326370 IC50 = 75.35 nM T31391 C30OEU 53326372 IC50 = 26.64 nM T31391 CL7T1U 53326374 IC50 = 33.78 nM T31391 CJP5V7 53326443 IC50 < 50000 nM T31391 C65JNF 53326490 IC50 > 50000 nM T31391 CYIA49 53326515 IC50 = 2.8 nM T31391 CV0H8P 53326691 IC50 = 110 nM T31391 C3ZWN6 53326704 IC50 = 100 nM T31391 C73SKG 53326705 IC50 = 1300 nM T31391 CG9V4W 53326706 IC50 = 110 nM T31391 C5K8CP 53326713 IC50 = 100 nM T31391 CHCE65 53326766 IC50 = 51 nM T31391 C4LCU1 53326767 IC50 = 1.2 nM T31391 C9UBW8 53326841 IC50 > 50000 nM T31391 C1HYV2 53326876 IC50 > 50000 nM T31391 CN12AO 53353383 IC50 = 255 nM T31391 C51GUC 53354365 IC50 = 67 nM T31391 CRJ5P9 53354369 IC50 = 102 nM T31391 C4G2HT 53354470 IC50 = 57 nM T31391 CUC1N3 53356519 Ki = 0.37 nM T31391 CSD1Q4 53357353 IC50 = 1.1 nM T31391 C5P9VZ 53465973 IC50 > 100000 nM T31391 C7OBF2 53465974 IC50 > 100000 nM T31391 CF5YJ8 53465975 IC50 > 100000 nM T31391 C5XER7 53466046 IC50 > 100000 nM T31391 CJ9T8M 53466047 IC50 > 50000 nM T31391 CP1CL8 53466049 IC50 > 100000 nM T31391 CPSQ16 53466050 IC50 > 100000 nM T31391 C4UC1P 53466119 IC50 > 100000 nM T31391 C59SML 53466121 IC50 > 100000 nM T31391 C7JPY2 53466122 IC50 > 100000 nM T31391 CYZK63 53466123 IC50 > 50000 nM T31391 CVJ0D5 53466193 IC50 > 100000 nM T31391 C2XE8Y 53466195 IC50 > 100000 nM T31391 C0P2YE 53466196 IC50 > 100000 nM T31391 CPA0K4 53466271 IC50 > 100000 nM T31391 CYG36O 53466361 IC50 = 17700 nM T31391 C5J9EB 53770701 IC50 = 510 nM T31391 CEK45S 54294055 IC50 = 87000 nM T31391 CRL42P 54573912 IC50 = 400 nM T31391 CUZS62 54580221 IC50 = 19 nM T31391 CG3S0X 54580222 IC50 = 0.7 nM T31391 CAQ8U7 54580310 IC50 = 21300 nM T31391 CX6K2C 54580311 IC50 = 26200 nM T31391 CS21IF 54580575 IC50 = 44.8 nM T31391 COZ98J 54580576 IC50 = 116 nM T31391 C2TSH1 54580577 IC50 = 54.1 nM T31391 CZL0N3 54580578 IC50 = 30.8 nM T31391 CNAQ35 54580579 IC50 = 7.4 nM T31391 CT24DU 54581222 IC50 = 7 nM T31391 CABF19 54581317 IC50 = 32700 nM T31391 C9JBG4 54581584 IC50 = 26.7 nM T31391 CJZ4S8 54582330 IC50 = 29100 nM T31391 C4L9SF 54582574 IC50 = 38.5 nM T31391 C0LQ9Z 54582575 IC50 = 13.7 nM T31391 CG84BL 54582898 IC50 = 12 nM T31391 CE5X6H 54583545 IC50 = 33.9 nM T31391 CB52YA 54583546 IC50 = 12 nM T31391 CST5M7 54584528 IC50 = 311 nM T31391 CV10YB 54585462 IC50 = 42.7 nM T31391 CG6M8J 54585463 IC50 = 38.9 nM T31391 CLCU50 54585464 IC50 = 1.3 nM T31391 CPWB63 54586434 IC50 = 50.7 nM T31391 C4G2PK 54586435 IC50 = 29 nM T31391 C71GKO 54586787 IC50 = 3 nM T31391 C4B2EW 54587461 IC50 = 92.6 nM T31391 C7VL9M 54587462 IC50 = 48.9 nM T31391 C04FAR 54587463 IC50 = 33.8 nM T31391 CQH56N 54698732 IC50 = 730 nM T31391 CY0ZH5 54698792 IC50 = 2950 nM T31391 C5UW0D 56652661 IC50 = 45 nM T31391 CMT0J9 56656630 IC50 = 133.6 nM T31391 C1QX0O 56657809 IC50 = 2 nM T31391 CU74VH 56658024 IC50 > 100000 nM T31391 CF6PV5 56658026 IC50 > 100000 nM T31391 C2KI8Y 56658028 IC50 > 100000 nM T31391 CY4E6U 56658138 IC50 > 100000 nM T31391 C5OT6W 56658248 IC50 = 26 nM T31391 C07KTW 56658249 IC50 > 1000 nM T31391 C1UDJ5 56659853 IC50 = 34 nM T31391 CX31TJ 56661748 IC50 = 0.34 nM T31391 COI5B0 56663604 IC50 = 65.1 nM T31391 C3VIA8 56663606 IC50 = 68.1 nM T31391 CD31AI 56663612 IC50 = 29.3 nM T31391 C52TBZ 56664349 IC50 = 20.4 nM T31391 C1PI4L 56664962 IC50 > 100000 nM T31391 C8GPO1 56665883 IC50 = 190 nM T31391 CA0BO6 56666264 IC50 > 100000 nM T31391 C8F5QV 56666543 IC50 = 4.2 nM T31391 C76MXW 56666747 IC50 = 49 nM T31391 C8DB0L 56670173 IC50 = 57 nM T31391 CJ9Q3V 56670497 IC50 = 47.8 nM T31391 CNL7D4 56671283 IC50 = 68.6 nM T31391 CXH5W7 56671896 IC50 > 100000 nM T31391 CMW3T8 56673186 IC50 > 100000 nM T31391 C1Q4XU 56673980 IC50 = 165.6 nM T31391 CP87EK 56674589 IC50 = 60.1 nM T31391 C2B6PY 56674700 IC50 = 34.8 nM T31391 C3OHT5 56675121 IC50 = 82.4 nM T31391 CBK31U 56675279 IC50 > 100000 nM T31391 CW8KU6 56675536 IC50 > 50000 nM T31391 C7WCK5 56676440 IC50 = 790 nM T31391 CH13RF 56676769 IC50 = 26 nM T31391 CX92YZ 56676772 IC50 = 2.7 nM T31391 CAO6M3 56677318 IC50 = 53.5 nM T31391 CPT94R 56678428 IC50 = 44.5 nM T31391 CN9S8A 56679836 IC50 > 100000 nM T31391 CF08YD 56680615 IC50 = 25.8 nM T31391 CZ1P7K 56851484 IC50 = 72 nM T31391 CU61OI 56851486 IC50 = 94 nM T31391 C9OL5C 56962798 IC50 = 10 nM T31391 CQX8J0 57385070 IC50 = 13.78 nM T31391 CPS89B 57385071 IC50 = 2.64 nM T31391 CNU9C0 57385072 IC50 = 2.34 nM T31391 CG5MT6 57385073 IC50 = 1.4 nM T31391 CQZ09L 57390626 IC50 = 80 nM T31391 CWR4E5 57390923 Ki = 0.55 nM T31391 C0RAD8 57390924 Ki = 0.3 nM T31391 C2AR3V 57391609 IC50 = 5.5 nM T31391 CKPB03 57391802 IC50 = 4 nM T31391 C8SW9E 57391803 IC50 = 10 nM T31391 C5UWC6 57391804 IC50 = 1 nM T31391 C78QEY 57391805 IC50 = 25 nM T31391 CYAQ83 57391806 IC50 = 20 nM T31391 COL58X 57391831 IC50 = 1 nM T31391 C5U6RF 57392407 IC50 = 13 nM T31391 CD0OT2 57392409 IC50 = 15 nM T31391 C4QYJ6 57392724 Ki = 0.27 nM T31391 CKS3X9 57393534 IC50 = 4 nM T31391 CM2EH0 57393535 IC50 = 250 nM T31391 CNP60T 57393564 IC50 = 10 nM T31391 CWDY79 57394441 Ki = 1.5 nM T31391 C5USX7 57395248 IC50 = 0.5 nM T31391 CJ80BU 57395249 IC50 = 1 nM T31391 C27MRL 57395273 IC50 = 20 nM T31391 CX5MG4 57395274 IC50 = 5 nM T31391 C40WGY 57395275 IC50 = 45 nM T31391 CZ23RJ 57395915 IC50 = 32 nM T31391 C8KMS2 57396206 Ki = 0.4 nM T31391 C0P8KM 57397016 IC50 = 2 nM T31391 CE85SV 57397017 IC50 = 2 nM T31391 C0J9MO 57397044 IC50 = 1 nM T31391 CCZ61A 57397045 IC50 = 8 nM T31391 CZJ1P7 57397046 IC50 = 9 nM T31391 C2QL6K 57397702 IC50 = 1.8 nM T31391 CBQ85O 57397704 IC50 = 11 nM T31391 C2ZE3R 57397706 IC50 = 28 nM T31391 CW97SN 57398006 Ki = 0.67 nM T31391 CSU2O9 57398779 IC50 = 2 nM T31391 C01KCU 57399665 Ki = 0.31 nM T31391 CDQ57A 57400458 IC50 = 3 nM T31391 CED9C4 57400459 IC50 = 2 nM T31391 CSEK63 57400487 IC50 = 4 nM T31391 CH6YT2 57400488 IC50 = 3 nM T31391 CX0N7O 57400489 IC50 = 60 nM T31391 C65ZFW 57401128 IC50 = 110 nM T31391 CYX43T 57401419 Ki = 0.29 nM T31391 CV2ME6 57402260 IC50 = 9 nM T31391 CQ1A8P 57402261 IC50 = 2 nM T31391 CW94QA 57402262 IC50 = 10 nM T31391 CMJA69 57402263 IC50 = 5 nM T31391 CV2CF5 57402294 IC50 = 23 nM T31391 C1T0AD 57403169 Ki = 0.43 nM T31391 C12QCM 57403170 Ki = 0.46 nM T31391 CX94UQ 57403171 Ki = 0.26 nM T31391 CX31VN 57403989 IC50 = 7.5 nM T31391 C4E7UI 57404016 IC50 = 2100 nM T31391 C5FHR8 57404017 IC50 = 15 nM T31391 C1L8YD 57404359 IC50 = 1650 nM T31391 C8SX7A 57404360 IC50 = 1100 nM T31391 C0Q1OZ 57404374 IC50 = 350 nM T31391 CXRS60 57406622 IC50 = 10 nM T31391 CNOX18 57406623 IC50 = 43.5 nM T31391 CZS03L 57406803 IC50 = 1.28 nM T31391 C80RBH 57406804 IC50 = 38.6 nM T31391 CMH17V 57406805 IC50 = 1.61 nM T31391 C2EX0S 57406806 IC50 = 19.3 nM T31391 CR6QP4 57406990 IC50 = 32 nM T31391 CFML71 57406991 IC50 = 8.15 nM T31391 C2PX9N 57406992 IC50 = 44.3 nM T31391 CHV47A 57406994 IC50 = 539 nM T31391 C0COE1 57407188 IC50 = 11.2 nM T31391 C5G3KT 57407189 IC50 = 9.31 nM T31391 C8MJK5 57407191 IC50 = 14.1 nM T31391 CVS34M 57407192 IC50 = 29.2 nM T31391 C7AZB3 57407370 IC50 = 82.2 nM T31391 CL0UA1 57525787 IC50 = 0.37 nM T31391 C75MLI 58874215 IC50 = 5.8 nM T31391 C9ZE7J 58874273 IC50 = 0.48 nM T31391 C3TSN9 58874353 IC50 = 14 nM T31391 C4KDJ8 58874386 IC50 = 0.55 nM T31391 COIQ05 58874405 IC50 = 418 nM T31391 C2I4JY 58874420 IC50 = 3.4 nM T31391 C0F5MP 58874435 IC50 = 4.8 nM T31391 CMW4N9 58874436 IC50 = 103 nM T31391 CZ4VD5 60032916 IC50 = 2.3 nM T31391 CI87CZ 61148520 Ki = 880 nM T31391 CAQ1O3 61148706 IC50 = 3.4 nM T31391 C68SUW 61174564 IC50 = 6.93 nM T31391 CXG48F 66545741 IC50 = 5.6 nM T31391 C2YPI7 66559296 IC50 = 0.61 nM T31391 CO2H1S 66559297 IC50 = 1.6 nM T31391 CRI16X 66559298 IC50 = 0.8 nM T31391 C5CX6V 66559299 IC50 = 0.59 nM T31391 CT15QA 66559300 IC50 = 0.39 nM T31391 CX48AY 66559301 IC50 = 1.2 nM T31391 CO0JP1 66559376 IC50 = 0.5 nM T31391 C2W0LI 66559377 IC50 = 0.55 nM T31391 C0NT6U 66559378 IC50 = 0.42 nM T31391 CG6EY9 66560524 IC50 = 0.61 nM T31391 CQMO80 66560608 IC50 = 0.73 nM T31391 CN4RL2 66560609 IC50 = 0.51 nM T31391 CS30FN 66560610 IC50 = 2.2 nM T31391 CZ4OU2 66560611 IC50 = 0.95 nM T31391 C02XCY 66560612 IC50 = 0.56 nM T31391 CW64RD 66561555 IC50 > 100000 nM T31391 C9GTI7 66561556 IC50 > 100000 nM T31391 CC85DI 66561873 IC50 = 2.3 nM T31391 C0QCA2 66561874 IC50 = 3.8 nM T31391 C5F6NR 66896083 Ki = 4 nM T31391 COIA16 66953432 IC50 = 645 nM T31391 C8CMU1 66953714 IC50 = 9 nM T31391 CUR3E1 66954220 IC50 = 1.6 nM T31391 CFW13I 66954232 IC50 = 100 nM T31391 CJY9L6 66962050 IC50 > 5000 nM T31391 CVOH80 66963065 IC50 = 290 nM T31391 CX7Z8R 67506840 IC50 = 4.5 nM T31391 C7Y1PN 67507142 IC50 = 4.3 nM T31391 CUIB42 67507176 IC50 = 0.2 nM T31391 CF92IB 67507913 IC50 = 0.26 nM T31391 C9SND1 68305755 IC50 > 100000 nM T31391 CP3E2X 68416066 IC50 = 0.3 nM T31391 CX34PR 68417107 IC50 = 0.94 nM T31391 CCS6K9 68417211 IC50 = 0.63 nM T31391 CUKP32 68417894 IC50 = 15 nM T31391 C54VZI 68417897 IC50 = 5 nM T31391 C69VWN 68418230 IC50 = 0.85 nM T31391 C6K0XY 68418986 IC50 = 3.4 nM T31391 C6U9SP 68419033 IC50 = 12 nM T31391 CFNU91 68419172 IC50 = 2.9 nM T31391 CZ7QX8 68419268 IC50 = 4 nM T31391 CEF87L 68419860 IC50 = 0.62 nM T31391 CH3Z7F 68658979 IC50 = 0.14 nM T31391 C31XFM 68828690 IC50 = 140 nM T31391 C7X2WD 68828739 IC50 = 100 nM T31391 C4C3BL 68828935 IC50 = 9.2 nM T31391 CR27HN 68829000 IC50 = 7.5 nM T31391 CVGE51 68829025 IC50 = 28 nM T31391 CU4K6C 68829197 IC50 = 55 nM T31391 CP1NA4 68829414 IC50 = 4.6 nM T31391 C45ICV 68829529 IC50 = 250 nM T31391 C06ZLV 68829605 IC50 = 720 nM T31391 C2K3PM 68829714 IC50 = 13 nM T31391 CZOG14 68829854 IC50 = 510 nM T31391 C6R7ZV 68829908 IC50 = 540 nM T31391 C5I4BK 68829917 IC50 = 620 nM T31391 CCE26Z 68830038 IC50 = 52 nM T31391 C1HR3S 68830304 IC50 = 17 nM T31391 C47PHV 68830457 IC50 = 170 nM T31391 CYV1A0 68830878 IC50 = 6.8 nM T31391 C62LNY 68830888 IC50 = 0.38 nM T31391 CL1VS3 68832119 IC50 = 630 nM T31391 C6HRX1 68845950 IC50 = 56 nM T31391 CDJI62 68914093 IC50 = 8.2 nM T31391 C2TOQ7 69089363 IC50 = 60000 nM T31391 CO95AZ 69442708 IC50 = 23 nM T31391 CY98ML 69445181 IC50 = 1.1 nM T31391 C6BR4W 69445419 IC50 = 30 nM T31391 CD42CX 69446073 IC50 = 29 nM T31391 CS85UC 69446132 IC50 = 470 nM T31391 CZ49VQ 69446166 IC50 = 3.7 nM T31391 CFL92T 69446285 IC50 = 80 nM T31391 CXM07R 69446326 IC50 = 87 nM T31391 CWTN63 69446993 IC50 = 17 nM T31391 CBQJ90 69447448 IC50 = 19 nM T31391 C67CPF 69576646 IC50 = 45.3 nM T31391 CW4O2C 69689410 Ki = 34 nM T31391 CQ2DM1 69890803 Ki = 910 nM T31391 C0C8JW 70293564 IC50 = 200 nM T31391 CK26FY 70295607 IC50 = 4 nM T31391 CV4X5S 70295927 IC50 = 7 nM T31391 CXSV41 70296244 IC50 = 3 nM T31391 C3SB1V 70296823 IC50 = 40 nM T31391 CL64SQ 70297489 IC50 = 19900 nM T31391 CXD5V6 70297609 IC50 = 2 nM T31391 CEG1L5 70330884 IC50 = 23 nM T31391 C5W6LY 70681316 IC50 = 14 nM T31391 CLO96S 70681357 IC50 > 100000 nM T31391 CWP41T 70681469 IC50 > 100000 nM T31391 C7Z2KY 70681470 IC50 > 100000 nM T31391 C97JFS 70682267 IC50 = 17 nM T31391 CE1FU2 70682268 IC50 = 17 nM T31391 CI8EQ5 70682492 IC50 = 45.3 nM T31391 C03SDB 70682493 IC50 = 67.7 nM T31391 CF0U3A 70682494 IC50 = 57.6 nM T31391 C8Z2UQ 70682495 IC50 = 57.4 nM T31391 C14AWU 70682667 IC50 = 31 nM T31391 C71BSM 70682668 IC50 = 723 nM T31391 C49RIG 70682669 IC50 = 14.3 nM T31391 C19XIQ 70683454 IC50 > 100000 nM T31391 C07ADL 70683455 IC50 > 100000 nM T31391 C4YW5T 70684349 IC50 = 200 nM T31391 C6W1CT 70684350 IC50 = 18000 nM T31391 C1GF3E 70684351 IC50 = 53 nM T31391 C2GUS0 70684568 IC50 = 212 nM T31391 CU1I5S 70684569 IC50 = 39 nM T31391 CM96VS 70684570 IC50 = 47.7 nM T31391 C1NHS4 70684571 IC50 = 42.2 nM T31391 C7HF3B 70684748 IC50 = 298 nM T31391 C74WUS 70684749 IC50 = 879 nM T31391 CL8OZ4 70684750 IC50 = 10.3 nM T31391 CV5T8O 70684751 IC50 = 13.2 nM T31391 CO2NK6 70685557 IC50 > 100000 nM T31391 CK0WX8 70685558 IC50 > 100000 nM T31391 CLF84U 70685559 IC50 > 100000 nM T31391 C0K7PS 70685560 IC50 > 100000 nM T31391 C2T0NS 70685696 IC50 > 100000 nM T31391 C1Q3ZO 70686506 IC50 = 6.2 nM T31391 CM90BQ 70686720 IC50 = 264 nM T31391 CNQ50W 70686721 IC50 = 569 nM T31391 CRA4G1 70686722 IC50 = 64.6 nM T31391 C5I9BL 70686723 IC50 = 24.9 nM T31391 CT2LK4 70686905 IC50 = 104 nM T31391 CVD76F 70687705 IC50 > 100000 nM T31391 C28GVW 70687706 IC50 > 100000 nM T31391 CLQC52 70688610 IC50 = 29 nM T31391 C6MZ4N 70688809 IC50 = 101 nM T31391 C3GY6A 70688810 IC50 = 103 nM T31391 CGQV87 70688811 IC50 = 31.2 nM T31391 CHL1T9 70688964 IC50 = 320 nM T31391 C76SEY 70688965 IC50 = 28 nM T31391 CDVF75 70688966 IC50 = 715 nM T31391 CK2UC9 70688967 IC50 = 869 nM T31391 CI0VF5 70688968 IC50 = 843 nM T31391 C8K4WF 70688969 IC50 = 74 nM T31391 CVYH31 70689717 IC50 = 23 nM T31391 CUY81P 70689750 IC50 > 100000 nM T31391 CX2O0Z 70689751 IC50 > 100000 nM T31391 C17YKW 70689752 IC50 > 100000 nM T31391 CYO5X6 70690674 IC50 = 59 nM T31391 C2J7FS 70690675 IC50 = 15 nM T31391 CL6KR9 70690676 IC50 = 0.3 nM T31391 CXE41O 70690893 IC50 = 30.5 nM T31391 C4QCP6 70691068 IC50 = 863 nM T31391 C7ROY0 70691069 IC50 = 100 nM T31391 CC0D7S 70691070 IC50 = 34 nM T31391 C87LMG 70691901 IC50 > 100000 nM T31391 CL5EG7 70691902 IC50 > 100000 nM T31391 CGND49 70691903 IC50 > 100000 nM T31391 CGT57B 70691904 IC50 > 100000 nM T31391 CT89CW 70691905 IC50 > 100000 nM T31391 C5WI6V 70691906 IC50 > 100000 nM T31391 C19FJC 70692822 IC50 = 48 nM T31391 C8JZ3Q 70692823 IC50 = 16 nM T31391 C7FIR6 70693034 IC50 = 85.7 nM T31391 CM3L1E 70693035 IC50 = 50.4 nM T31391 C3DV6C 70693036 IC50 = 56.4 nM T31391 C3MF7C 70693037 IC50 = 91.5 nM T31391 C5YQ9B 70693038 IC50 = 33.9 nM T31391 CEQ4N8 70693039 IC50 = 76.2 nM T31391 CYQO06 70693040 IC50 = 36.7 nM T31391 C0S9LO 70693199 IC50 = 890 nM T31391 CY7M8K 70693200 IC50 = 19 nM T31391 C4P5TC 70693201 IC50 = 863 nM T31391 CEB6L2 70693202 IC50 = 116 nM T31391 CQMV53 70693949 IC50 > 100000 nM T31391 CBP8U7 70693950 IC50 > 100000 nM T31391 C0I2CV 70693951 IC50 > 100000 nM T31391 CCB64G 70693952 IC50 > 100000 nM T31391 C3ZUK2 70693953 IC50 > 100000 nM T31391 CS76EN 70693954 IC50 > 100000 nM T31391 C27PFC 70693955 IC50 > 100000 nM T31391 CVY48R 70693956 IC50 > 100000 nM T31391 CIX3F9 70694853 IC50 = 6.5 nM T31391 CQJD92 70694854 IC50 = 20 nM T31391 C8JRC5 70695073 IC50 = 99.7 nM T31391 CA0W8R 70695074 IC50 = 65.4 nM T31391 CYB1P3 70695075 IC50 = 74.4 nM T31391 C4ETL9 70695076 IC50 = 113.9 nM T31391 C5ZN7P 70695277 IC50 = 107 nM T31391 C3S5EX 70695278 IC50 = 26 nM T31391 CC6B7L 70695279 IC50 = 694 nM T31391 CXG5O4 70695280 IC50 = 311 nM T31391 CA01KO 70696068 IC50 > 100000 nM T31391 CSW43K 70696069 IC50 = 13100 nM T31391 C1NGL5 70696903 IC50 = 2.1 nM T31391 CR6FY8 70697121 IC50 = 194 nM T31391 C2B5UF 70697122 IC50 = 291 nM T31391 CV38GW 70697123 IC50 = 52.6 nM T31391 CJ4M0N 70697124 IC50 = 50.6 nM T31391 C4GIH1 70697292 IC50 = 31 nM T31391 CALB67 70697293 IC50 = 11.6 nM T31391 C19ZWC 70789754 IC50 > 100000 nM T31391 C31UTS 71184301 IC50 = 250 nM T31391 C8LY1U 71184352 IC50 = 9 nM T31391 C9IRW7 71184590 IC50 = 40 nM T31391 C8BK4O 71184607 IC50 = 4200 nM T31391 CS29MW 71184623 IC50 = 15700 nM T31391 C08NDK 71184749 IC50 = 20 nM T31391 CP91OE 71203742 IC50 = 625 nM T31391 CP6G5W 71203746 IC50 = 11.2 nM T31391 C32UMV 71203748 IC50 = 1.7 nM T31391 C04XQY 71203752 IC50 = 27.4 nM T31391 CE2I0K 71203758 IC50 = 123 nM T31391 CIQ7O2 71203767 IC50 = 13.5 nM T31391 C5GEJ9 71203769 IC50 = 156.1 nM T31391 C7LKV0 71203783 IC50 = 10.6 nM T31391 CBK26E 71449262 IC50 = 160 nM T31391 CW8JE0 71449264 IC50 = 150 nM T31391 CD9C3R 71449266 IC50 = 6900 nM T31391 CBX46U 71449270 IC50 = 54 nM T31391 CT35BK 71449272 IC50 = 64 nM T31391 C6D0WY 71449276 IC50 = 22 nM T31391 C46QSR 71449278 IC50 = 660 nM T31391 CKR1E6 71449280 IC50 = 72 nM T31391 CAJ8F0 71449608 IC50 = 20 nM T31391 CM5DB6 71450086 IC50 > 100000 nM T31391 CQU0Z1 71450087 IC50 > 100000 nM T31391 C65BCE 71450089 IC50 > 100000 nM T31391 CP9K2W 71450603 IC50 = 12 nM T31391 C8GBF1 71450604 IC50 = 670 nM T31391 CA3LP4 71450605 IC50 = 94 nM T31391 CD80JE 71451064 IC50 = 90 nM T31391 CH83NV 71451066 IC50 = 13 nM T31391 CM86TF 71451071 IC50 = 400 nM T31391 C9BK1J 71451073 IC50 = 17 nM T31391 CLC2N8 71451900 IC50 > 100000 nM T31391 CMU63C 71451901 IC50 > 100000 nM T31391 CT5WU4 71451902 IC50 > 100000 nM T31391 CL0X3F 71451939 IC50 > 100000 nM T31391 C7ZN6W 71452445 IC50 = 41 nM T31391 CKVA72 71452446 IC50 = 250 nM T31391 CP5NS6 71452447 IC50 = 110 nM T31391 C61LNR 71452448 IC50 = 83 nM T31391 C2J3GF 71452890 IC50 > 10000 nM T31391 C4GQ5B 71452892 IC50 = 90 nM T31391 CEM2O9 71453723 IC50 > 100000 nM T31391 CB1EX7 71453762 IC50 > 100000 nM T31391 CN4FE7 71454208 IC50 = 24 nM T31391 CD4IE2 71454659 IC50 = 3500 nM T31391 C2GO8L 71454668 IC50 = 12 nM T31391 CT9YS3 71454883 IC50 = 16 nM T31391 CBOK64 71455456 IC50 > 100000 nM T31391 CD32GT 71455458 IC50 > 100000 nM T31391 CQA9L7 71455494 IC50 > 100000 nM T31391 C1LRH5 71455960 IC50 = 84 nM T31391 CGH7R6 71455961 IC50 = 55 nM T31391 CGKJ82 71456385 IC50 = 38 nM T31391 CCY8P7 71456387 IC50 = 8900 nM T31391 CIC59O 71456389 IC50 = 3.8 nM T31391 CNGO29 71456391 IC50 = 60 nM T31391 C7AU4I 71456393 IC50 = 17 nM T31391 CVIF92 71456398 IC50 > 10000 nM T31391 C0CHQ9 71456400 IC50 = 66 nM T31391 C4T7CO 71457236 IC50 > 100000 nM T31391 C3GAO1 71457237 IC50 > 100000 nM T31391 CE3MP2 71457238 IC50 > 100000 nM T31391 C42BSO 71457239 IC50 > 100000 nM T31391 C8VI9L 71457240 IC50 > 50000 nM T31391 CK0O9D 71457760 IC50 = 490 nM T31391 C59TGZ 71457761 IC50 = 16 nM T31391 C8O6HJ 71457762 IC50 = 59 nM T31391 CBKA19 71457763 IC50 = 190 nM T31391 CI15BH 71457764 IC50 = 160 nM T31391 C5T6QP 71457765 IC50 = 72 nM T31391 C87VPZ 71458224 IC50 = 51 nM T31391 C89DPI 71458226 IC50 = 10 nM T31391 CK6S7X 71458227 IC50 = 6.3 nM T31391 CB67AV 71458229 IC50 = 3.5 nM T31391 CLRE92 71458241 IC50 = 66 nM T31391 CW76HL 71458243 IC50 = 16 nM T31391 CIO50T 71459090 IC50 > 100000 nM T31391 CXIM97 71459091 IC50 > 100000 nM T31391 CJ6N1C 71459092 IC50 > 100000 nM T31391 CUB4V8 71459679 IC50 = 7.8 nM T31391 C10JPO 71459680 IC50 = 330 nM T31391 CWQ59G 71460084 IC50 = 25 nM T31391 CZ7E1K 71460086 IC50 = 56 nM T31391 CS89OV 71460088 IC50 = 21 nM T31391 C6Z8RT 71460094 IC50 = 271 nM T31391 CKXG80 71460143 IC50 = 0.32 nM T31391 CEY13Z 71460148 IC50 = 6.3 nM T31391 CEU0B1 71460149 IC50 > 1000 nM T31391 CSC3I7 71460901 IC50 > 100000 nM T31391 CG7VX2 71460902 IC50 > 100000 nM T31391 C5K3WJ 71460903 IC50 > 100000 nM T31391 C3UF9P 71460904 IC50 > 100000 nM T31391 CUJT52 71461398 IC50 = 1100 nM T31391 CQ6GA0 71461399 IC50 = 50 nM T31391 CJ07GY 71461805 IC50 = 110 nM T31391 C8LB7A 71461808 IC50 = 11 nM T31391 C79EIW 71461811 IC50 = 1.6 nM T31391 CPAN79 71461821 IC50 = 3400 nM T31391 C02ALK 71461822 IC50 = 340 nM T31391 C7TS9F 71462596 IC50 > 100000 nM T31391 C63SUR 71462597 IC50 > 100000 nM T31391 CZT3S0 71462641 IC50 > 100000 nM T31391 CY2W5V 71463119 IC50 = 390 nM T31391 C16PTB 71463120 IC50 = 280 nM T31391 CKZ17B 71463121 IC50 = 60 nM T31391 C4VKM3 71463122 IC50 = 100 nM T31391 CY4W8D 71520057 IC50 = 660 nM T31391 C0JUM4 71520123 IC50 = 1320 nM T31391 CZ0UG8 71520163 IC50 = 720 nM T31391 CQO90M 71550930 IC50 = 1.55 nM T31391 C57JVN 71566829 Ki = 4 nM T31391 CMX9E3 71566830 Ki = 18 nM T31391 CDJ2T7 71566831 Ki = 14 nM T31391 C2SB3J 71566832 Ki = 18 nM T31391 C3J4DA 71566833 Ki = 11 nM T31391 CGVS23 71566834 Ki = 18 nM T31391 C5EQ8X 71566966 Ki = 13 nM T31391 C1VG2P 71566967 Ki = 30 nM T31391 C8FH4K 71566968 Ki = 8 nM T31391 C6AQ8P 71566969 Ki = 5 nM T31391 CM3NB6 71566970 Ki = 4 nM T31391 C92TKQ 71566971 Ki = 2 nM T31391 CZN30Q 71567105 Ki = 35 nM T31391 CL0BY5 71567106 Ki = 38 nM T31391 C63UAJ 71567107 Ki = 15 nM T31391 CPLH40 71567235 Ki = 10 nM T31391 CNM83T 71568676 Ki = 98 nM T31391 CEGB81 71568801 Ki = 75 nM T31391 C1G5WV 71568802 Ki = 25 nM T31391 CGXB93 71568803 Ki = 23 nM T31391 C0XK9O 71568804 Ki = 18 nM T31391 CL57TN 71568805 Ki = 14 nM T31391 CGJQ86 71568806 Ki = 18 nM T31391 CY3ZG6 71582959 IC50 = 211.9 nM T31391 C97MES 71583061 IC50 = 44 nM T31391 CB1YX0 71583062 IC50 = 44.1 nM T31391 CX43IU 71583063 IC50 = 27.6 nM T31391 C3KW9P 71583064 IC50 = 48.2 nM T31391 CEK26O 71583065 IC50 = 7.05 nM T31391 C53UMG 71583066 IC50 = 139.2 nM T31391 C9IRB0 71583175 IC50 = 60.1 nM T31391 CY87XJ 71583176 IC50 = 14.5 nM T31391 CD5O8F 71583177 IC50 = 52.6 nM T31391 C85BGF 71583178 IC50 = 11.4 nM T31391 CA67NL 71583179 IC50 = 4.67 nM T31391 C17-APR 71583292 IC50 = 5.93 nM T31391 CUH48W 71583293 IC50 = 15.5 nM T31391 C9AKS7 71594483 IC50 = 22390 nM T31391 C7B8AO 71621488 IC50 > 100000 nM T31391 C8T2PW 71655265 IC50 = 2800 nM T31391 CVB75Q 71655394 IC50 = 1800 nM T31391 CH4ZS0 71655395 IC50 > 100000 nM T31391 CC93KJ 71655554 IC50 > 100000 nM T31391 CN90KH 71655555 IC50 > 100000 nM T31391 CUT37D 71655556 IC50 > 100000 nM T31391 C71OFQ 71655557 IC50 > 100000 nM T31391 C7R6HU 71655622 IC50 > 100000 nM T31391 C2NA1M 71655623 IC50 > 100000 nM T31391 CDF08H 71655624 IC50 > 100000 nM T31391 CBEX27 71655625 IC50 > 100000 nM T31391 CT6XB5 71655626 IC50 > 100000 nM T31391 C1ND2P 71655627 IC50 > 100000 nM T31391 CXZ8N4 71667081 IC50 > 100000 nM T31391 CJ9QU7 71667226 IC50 > 100000 nM T31391 CE0Z8G 71667227 IC50 > 100000 nM T31391 CL7CS3 71667230 IC50 > 100000 nM T31391 CB6SI5 71667231 IC50 > 100000 nM T31391 C75UWV 71667375 IC50 > 100000 nM T31391 C19CTI 71667376 IC50 > 100000 nM T31391 C69CJB 71667378 IC50 > 100000 nM T31391 C07HNK 71667379 IC50 > 100000 nM T31391 CK74SP 71667380 IC50 > 100000 nM T31391 CMYZ68 71667381 IC50 > 100000 nM T31391 CDI39U 71667510 IC50 > 100000 nM T31391 CT49CO 71674688 IC50 = 34650 nM T31391 C8YTW3 71716406 Ki = 109 nM T31391 CQR5A1 71718946 IC50 = 460 nM T31391 CXKP89 71719452 Ki = 695 nM T31391 C0V3ZW 71720156 IC50 = 860 nM T31391 C0SC3Q 71720681 Ki = 1201 nM T31391 C7BD2R 71720854 IC50 = 2 nM T31391 CW3JG7 71731241 IC50 > 10000 nM T31391 C3D4HJ 71731243 IC50 = 31.3 nM T31391 CU6BC5 71731355 IC50 = 22 nM T31391 C5TS9Y 71731356 IC50 = 3.1 nM T31391 C5RTY9 71731357 IC50 = 3.4 nM T31391 CD9F5X 71731476 IC50 = 10.8 nM T31391 C3IO9H 71731477 IC50 = 6.6 nM T31391 CVAD62 71731478 IC50 = 2 nM T31391 C1ON0X 71731479 IC50 = 9.1 nM T31391 CZYQ05 71731604 IC50 = 1.9 nM T31391 C40YRO 71731605 IC50 = 0.7 nM T31391 C9Q8MO 72164809 IC50 = 9.39 nM T31391 CL5X1Z 72164811 IC50 = 25.5 nM T31391 C7N8WB 72164813 IC50 = 17.61 nM T31391 C2R0NV 72164815 IC50 = 8.28 nM T31391 C4JLM5 72164817 IC50 = 19.54 nM T31391 C6RQ9A 72164819 IC50 = 7.56 nM T31391 C38GWP 72164942 IC50 = 3.79 nM T31391 C4T0MY 72164944 IC50 = 15.24 nM T31391 C0T4UW 72164946 IC50 = 10.45 nM T31391 CLV02R 72164948 IC50 = 6.05 nM T31391 CHPN10 72164950 IC50 = 20.84 nM T31391 CI78FQ 72165082 IC50 = 7.5 nM T31391 CN0VU2 72165084 IC50 = 4.35 nM T31391 C84SYX 72165086 IC50 = 8.57 nM T31391 C1RQA3 72165088 IC50 = 10.02 nM T31391 CH51ZR 72165090 IC50 = 15.7 nM T31391 C1HL2A 72188903 IC50 = 13100 nM T31391 CLS1A0 72188904 IC50 > 100000 nM T31391 CO15AV 72188905 IC50 = 0.66 nM T31391 CPDC28 72188906 IC50 = 140 nM T31391 CL7P3D 72193502 IC50 = 24400 nM T31391 C4AXB8 72193503 IC50 = 38000 nM T31391 CQC28P 72193504 IC50 = 2800 nM T31391 CV87PE 72193505 IC50 = 26600 nM T31391 C65DFP 72697059 IC50 = 18 nM T31391 CX07OC 72697060 IC50 = 248 nM T31391 CZ56DO 72697061 IC50 = 11 nM T31391 C1A2KX 72697062 IC50 = 17 nM T31391 CS5U1F 72697063 IC50 = 29 nM T31391 CA3HI1 72697064 IC50 = 75 nM T31391 CCZJ47 72697206 IC50 = 20 nM T31391 CWNZ91 72697207 IC50 = 21 nM T31391 C6BWI4 72697208 IC50 = 31 nM T31391 C9JA1Q 72697209 IC50 = 4 nM T31391 CF6A8N 72697210 IC50 = 4 nM T31391 CTMR03 72697211 IC50 = 42 nM T31391 CP9NV5 72697212 IC50 = 27 nM T31391 C1P8HS 72697352 IC50 = 46 nM T31391 CC7G3M 72697353 IC50 = 63 nM T31391 CXYO73 72697354 IC50 = 209 nM T31391 CAXV78 72697355 IC50 = 17 nM T31391 CGV09W 72697356 IC50 = 3 nM T31391 CIF9D7 72697357 IC50 = 4 nM T31391 CC8RA6 72697358 IC50 = 15 nM T31391 C1EC7S 72697359 IC50 = 292 nM T31391 C8CRO6 72697494 IC50 = 5 nM T31391 C03NKY 72697495 IC50 = 6 nM T31391 CP0MU3 72697496 IC50 = 125 nM T31391 CI60AK 72697497 IC50 = 94 nM T31391 CO19YK 72697498 IC50 = 22 nM T31391 C47IGZ 72697499 IC50 = 20 nM T31391 C65OPG 72697500 IC50 = 6 nM T31391 C3ZP7N 72697501 IC50 = 23 nM T31391 C7EF8C 72697646 IC50 = 60 nM T31391 C08IGP 72699737 IC50 = 1.98 nM T31391 CMT61I 72707535 IC50 = 198 nM T31391 CAEF04 72707536 IC50 = 2177.5 nM T31391 C7ARW4 72707537 IC50 = 1.2 nM T31391 C8D5PB 72725804 IC50 = 11900 nM T31391 CC10AZ 73345857 IC50 > 100000 nM T31391 CSZR98 73346173 IC50 = 48 nM T31391 C1L4RX 73346174 IC50 = 1 nM T31391 CX4F0Y 73347359 IC50 > 100000 nM T31391 C3XFM5 73347360 IC50 > 100000 nM T31391 CGNL10 73347698 IC50 = 720 nM T31391 CR09PJ 73348871 IC50 > 10000 nM T31391 CA79DR 73349143 IC50 = 265 nM T31391 CO5TB8 73349220 IC50 = 37 nM T31391 C06WRM 73350448 IC50 > 100000 nM T31391 C1T7LK 73350449 IC50 > 100000 nM T31391 CCIZ12 73350450 IC50 > 100000 nM T31391 CNC6B8 73350798 IC50 = 125 nM T31391 CDBV29 73350799 IC50 = 27 nM T31391 CYG04J 73352283 IC50 = 12600 nM T31391 CFV5U3 73353424 IC50 > 100000 nM T31391 CRS4O0 73353425 IC50 > 100000 nM T31391 C7X9ZG 73353601 IC50 > 1000 nM T31391 CV6BA3 73353756 IC50 = 37 nM T31391 C51QGP 73353757 IC50 = 27 nM T31391 CBK37N 73353758 IC50 = 64 nM T31391 CLYP23 73354936 IC50 > 100000 nM T31391 CLO76J 73355285 IC50 = 11 nM T31391 CCVT96 73355286 IC50 = 1.6 nM T31391 CH9W2R 73356494 IC50 > 100000 nM T31391 CKD46T 73356495 IC50 > 100000 nM T31391 CI0N6E 73356496 IC50 > 10000 nM T31391 C7R3ZT 76309823 Ki = 142000 nM T31391 CY0N9K 76311138 IC50 = 170 nM T31391 CWK7M6 76311139 IC50 = 50 nM T31391 CF5S9X 76313540 Ki = 61000 nM T31391 CIP4R0 76314754 IC50 = 40 nM T31391 C3HRA1 76314755 IC50 = 50 nM T31391 C1ZAC3 76317994 IC50 = 113760 nM T31391 C68JOX 76318341 IC50 = 30 nM T31391 CET31O 76318342 Ki = 3.5 nM T31391 CP0H8I 76320760 Ki = 4500 nM T31391 C9UGA3 76325642 IC50 = 113600 nM T31391 CNIP02 76325643 IC50 = 5 nM T31391 C08DYM 76325644 IC50 = 120 nM T31391 C3C7HE 76325645 Ki = 9 nM T31391 CWBL62 76327979 Ki = 6300 nM T31391 CW4M6E 76329221 IC50 = 390 nM T31391 C3LPR2 76331631 Ki = 5000 nM T31391 C7S6EY 76332265 IC50 = 4364 nM T31391 CH95ZJ 76336484 IC50 = 520 nM T31391 C4W7RE 77461184 IC50 = 8.5 nM T31391 CRG30N 86267497 IC50 = 148 nM T31391 C7JRH1 86267498 IC50 = 89.6 nM T31391 CTXI04 86267501 IC50 = 3 nM T31391 CO78UK 86267502 IC50 = 3.4 nM T31391 C7K2NA 86267708 IC50 = 3.8 nM T31391 CPS4U2 86268135 IC50 = 2290 nM T31391 C9GA1T 86268138 IC50 = 299 nM T31391 CBJ6N8 86268336 IC50 = 19.2 nM T31391 CA3L2Q 86268337 IC50 = 15.4 nM T31391 C6HCF9 86268525 IC50 = 18.6 nM T31391 CLG83C 86268944 IC50 = 4.9 nM T31391 C31OGJ 86279928 IC50 = 10.8 nM T31391 CB60OP 89488720 IC50 = 2.6 nM T31391 CIV7Y8 89668929 IC50 > 100000 nM T31391 C87GJT 89704940 IC50 > 100000 nM T31391 CHI7U9 89704942 IC50 > 100000 nM T31391 CSLI09 89704955 IC50 > 100000 nM T31391 CA3K7R 89704970 IC50 > 100000 nM T31391 CF89OD 89705045 IC50 > 100000 nM T31391 CK3Z8J 89705076 IC50 > 100000 nM T31391 CH6P0S 89705081 IC50 > 100000 nM T31391 C63DGS 89705096 IC50 > 100000 nM T31391 CND56S 89705098 IC50 > 100000 nM T31391 C0CKQ7 89705100 IC50 > 100000 nM T31391 C0CPD1 89705103 IC50 > 100000 nM T31391 C1IL7N 89705109 IC50 > 50000 nM T31391 CA48MR 89705136 IC50 > 100000 nM T31391 C5F9OA 89705152 IC50 > 100000 nM T31391 C1VSG5 89705179 IC50 > 100000 nM T31391 CHAS49 89705195 IC50 > 100000 nM T31391 C0RP1J 89705223 IC50 > 100000 nM T31391 CQO0I6 89705242 IC50 > 100000 nM T31391 C7DF1P 89705244 IC50 > 100000 nM T31391 C03OGJ 89705273 IC50 > 100000 nM T31391 CGX4I7 89705275 IC50 = 19000 nM T31391 CX9BC3 89712515 IC50 > 100000 nM T31391 CM5N8H 90654714 IC50 = 1436 nM T31391 CFY63H 90654715 IC50 = 378 nM T31391 CC6VX3 90654716 IC50 = 382 nM T31391 CA0SL5 90654717 IC50 = 342 nM T31391 CAM68Q 90654718 IC50 = 217 nM T31391 CQ93MA 90654719 IC50 = 193 nM T31391 CNDG24 90654720 IC50 = 1388 nM T31391 CC46WF 90654721 IC50 = 452 nM T31391 CCX20I 90654722 IC50 = 443 nM T31391 COV32D 90654723 IC50 = 404 nM T31391 CZ7KU8 90654724 IC50 = 885 nM T31391 CUH0W7 90654725 IC50 = 910 nM T31391 CCX14G 90654726 IC50 = 1034 nM T31391 CXUY06 90654727 IC50 = 1023 nM T31391 CKC94W 90654728 IC50 = 997 nM T31391 C8VBP2 90654729 IC50 = 119 nM T31391 C2UN8K 90654730 IC50 = 84 nM T31391 C1GSQ3 90654731 IC50 = 77.6 nM T31391 C47YVG 90654732 IC50 = 122 nM T31391 C20CDE 90654733 IC50 = 79 nM T31391 C9B2MJ 90654734 IC50 = 74 nM T31391 C30OWT 90654735 IC50 = 157 nM T31391 C3XP8C 90654736 IC50 = 119 nM T31391 CQD53I 90654737 IC50 = 125 nM T31391 C10TVX 90654738 IC50 = 111 nM T31391 C17RCY 90654739 IC50 = 19 nM T31391 CLT2X9 90654740 IC50 = 197 nM T31391 CDO0J4 90654741 IC50 = 148 nM T31391 CS62OC 90654742 IC50 = 134 nM T31391 C4B8KC 90654743 IC50 = 137 nM T31391 CKU5M8 90654744 IC50 = 43 nM T31391 C6TGZ5 90655538 IC50 > 100000 nM T31391 C9P3HJ 90655539 IC50 > 100000 nM T31391 CT98OM 90655540 IC50 > 100000 nM T31391 CVQ8M4 90655541 IC50 > 100000 nM T31391 CT6Q2L 90655542 IC50 > 100000 nM T31391 C7Z4GV 90655543 IC50 > 100000 nM T31391 CE3HC2 90655544 IC50 > 100000 nM T31391 CU2I3V 90655545 IC50 > 100000 nM T31391 C2NZ7X 90655546 IC50 > 100000 nM T31391 C0E5UP 90655547 IC50 > 100000 nM T31391 CF23RI 90655548 IC50 > 100000 nM T31391 CW3QG7 90655549 IC50 > 100000 nM T31391 CHG4E2 90655550 IC50 > 100000 nM T31391 CTA78W 90655551 IC50 > 100000 nM T31391 CA6S4W 90655552 IC50 > 100000 nM T31391 C3LT0S 90655553 IC50 > 100000 nM T31391 CEW45X 90655554 IC50 > 100000 nM T31391 CRX52D 90655555 IC50 > 100000 nM T31391 C9KG1U 90655556 IC50 > 100000 nM T31391 CXYE76 90655557 IC50 > 100000 nM T31391 CES85Q 90655558 IC50 > 100000 nM T31391 CK7IB9 90655559 IC50 >= 100000 nM T31391 CAG5X4 90655560 IC50 > 100000 nM T31391 C3IJA0 90655561 IC50 > 100000 nM T31391 C4V0ZY 90655562 IC50 > 100000 nM T31391 CY9G8Q 90655563 IC50 > 100000 nM T31391 CPIN84 90664318 IC50 = 53 nM T31391 CY76CR 90664436 IC50 = 1.8 nM T31391 C8YPL7 90664437 IC50 = 11 nM T31391 CU9LB2 90664438 IC50 > 100000 nM T31391 CQ20XA 90664578 IC50 > 100000 nM T31391 CV87ZH 90664579 IC50 > 100000 nM T31391 C9OC4Q 90664688 IC50 = 8.1 nM T31391 CJVF52 90664689 IC50 = 19 nM T31391 CDEN13 90664693 IC50 > 100000 nM T31391 CFG21I 90664805 IC50 = 2.9 nM T31391 C37YWE 90664828 IC50 = 84 nM T31391 CP60NA 90664941 IC50 = 7.8 nM T31391 CJ04US 90664942 IC50 = 69 nM T31391 CCH31U 90665060 IC50 = 23 nM T31391 C4LB2V 90665061 IC50 = 17 nM T31391 C0C1VT 90665186 IC50 = 12 nM T31391 CJ81VK 90665187 IC50 = 73 nM T31391 CHB2D6 90666864 IC50 = 16580 nM T31391 CFH71J 91937923 IC50 = 3730 nM T31391 COA7Z6 92131131 IC50 = 14 nM T31391 CBQ38C 101879512 IC50 = 170 nM T31391 CM7E4V 101887269 IC50 > 50000 nM T31391 C8EH0J 101887270 IC50 = 5.8 nM T31391 CDT67J 101887271 IC50 = 25 nM T31391 C4F2CS 101887272 IC50 > 100000 nM T31391 C58XWA 101887273 IC50 = 18100 nM T31391 C3Y9ET 101887274 IC50 > 100000 nM T31391 C1AF8C 101887275 IC50 = 1440 nM T31391 CH7QC5 101887276 IC50 > 50000 nM T31391 CO4FR2 101887277 IC50 = 29 nM T31391 C9JEH0 101887278 IC50 = 13900 nM T31391 C52GIO 101887279 IC50 > 100000 nM T31391 CO95EZ 118705501 IC50 = 570 nM T31391 CH8VO2 118705502 IC50 = 30 nM T31391 CZ1G3O 118712516 IC50 > 100000 nM T31391 C8X4JA 118712517 IC50 > 100000 nM T31391 CC29AB 118712518 IC50 > 100000 nM T31391 CB09PD 118712519 IC50 > 100000 nM T31391 CD4U1X 118712520 IC50 > 100000 nM T31391 CU0V5J 118712521 IC50 > 100000 nM T31391 C03OUP 118712522 IC50 > 100000 nM T31391 CT2MZ8 118712764 IC50 = 450 nM T31391 C3W5RU 118712765 IC50 = 220 nM T31391 CKA1N5 118712766 IC50 = 160 nM T31391 C8M6ZW 118712767 IC50 = 220 nM T31391 CV5C6D 118712768 IC50 = 320 nM T31391 C2NSC7 118712769 IC50 = 430 nM T31391 CV8JY3 118712770 IC50 = 640 nM T31391 C4KCZ1 118712771 IC50 = 770 nM T31391 CAR4W5 118712772 IC50 = 40 nM T31391 CRWT85 118712773 IC50 = 530 nM T31391 C36YUB 118712774 IC50 = 1580 nM T31391 C4T2FY 118712775 IC50 = 50 nM T31391 C0MYA1 118712776 IC50 = 1940 nM T31391 C8IF4E 118712777 IC50 = 440 nM T31391 CJ8EL0 118712778 IC50 = 70 nM T31391 C07UOL 118712779 IC50 = 360 nM T31391 C25HYG 118712780 IC50 = 130 nM T31391 CD0HQ4 118712781 IC50 = 270 nM T31391 C5D9RH 118712782 IC50 = 8800 nM T31391 CB7NX6 118712783 IC50 = 1980 nM T31391 C46TMQ 118712785 IC50 = 70 nM T31391 CA1I4M 118712786 IC50 = 47440 nM T31391 CUN79Q 118712787 IC50 = 9650 nM T31391 C5M3BX 118712788 IC50 = 10 nM T31391 CV3AK9 118717414 IC50 = 2390 nM T31391 C1NAQ9 118717415 IC50 > 100000 nM T31391 CKES65 118717416 IC50 > 100000 nM T31391 CYP07B 118719171 Ki = 6000 nM T31391 CD3L8W 118719172 Ki = 520 nM T31391 C8WJL2 118719173 Ki = 900 nM T31391 C5HU8M 118719174 Ki = 2700 nM T31391 C36XYR 118722404 IC50 = 5810 nM T31391 CX6J2E 118722405 IC50 = 340 nM T31391 C7BD8K 118722406 IC50 = 380 nM T31391 C0K6YG 118722407 IC50 = 760 nM T31391 CK7HN4 118722408 IC50 = 70 nM T31391 CFV6N4 118722409 IC50 = 3660 nM T31391 CK71WT 118722410 IC50 = 70 nM T31391 CI74ZM 118722411 IC50 = 80 nM T31391 CH1P7Y 118722412 IC50 = 70 nM T31391 CL8TY5 118722413 IC50 = 180 nM T31391 CGK98I 118722414 IC50 = 320 nM T31391 CBK91L 118722415 IC50 = 510 nM T31391 C8KUP0 118722416 IC50 = 290 nM T31391 C76DBO 118722417 IC50 = 540 nM T31391 CW6L5X 118722418 IC50 = 330 nM T31391 CM6Y5I 118722419 IC50 = 430 nM T31391 C37BGF 118722420 IC50 = 610 nM T31391 COG4V6 118722421 IC50 = 140 nM T31391 CIQ5Z7 118722422 IC50 = 430 nM T31391 CH6GX2 118728164 IC50 = 6 nM T31391 CFCI13 118728166 IC50 = 4.7 nM T31391 CS08AG 118728168 IC50 = 1.4 nM T31391 C0AG2Q 118728920 IC50 = 500 nM T31391 CE1ZS2 118728922 IC50 = 230 nM T31391 CVG84E 118728927 IC50 = 640 nM T31391 CBI68Y 118728931 IC50 = 36 nM T31391 CI0E1U 118736611 IC50 = 695 nM T31391 C2NX7C 118736612 IC50 = 2801 nM T31391 CP71VU 118736613 IC50 = 27.54 nM T31391 CL40TU 118736614 IC50 = 145 nM T31391 CJI2B8 118736615 IC50 = 85 nM T31391 C15XMK 118736616 IC50 = 108 nM T31391 C1IGJ6 118736617 IC50 = 67 nM T31391 C4BI2T 118736618 IC50 = 258 nM T31391 CED50R 118736620 IC50 = 100 nM T31391 C3DT9O 118736622 IC50 = 94 nM T31391 C6TYS7 122172854 IC50 = 4376 nM T31391 C2U5PE 122178432 IC50 = 20 nM T31391 C7TEY3 122178433 IC50 = 19.8 nM T31391 C8OLP9 122178434 IC50 = 346 nM T31391 C9GP3L 122178435 IC50 = 2.9 nM T31391 C8P2DB 122178436 IC50 = 6.4 nM T31391 CGFU89 122178437 IC50 = 3.4 nM T31391 CN78TQ 122189864 IC50 = 650 nM T31391 CNM82F 122189865 IC50 > 100000 nM T31391 C19GHJ 122189866 IC50 = 12200 nM T31391 C3U9KC 122189867 IC50 > 100000 nM T31391 CW5V3U 122189868 IC50 = 180 nM T31391 CCG05R 122189869 IC50 = 1800 nM T31391 CI01PT 122189870 IC50 = 180 nM T31391 C80EWF 122189871 IC50 = 220 nM T31391 C3N7JC 122189872 IC50 > 100000 nM T31391 CG8O1J 122189873 IC50 > 100000 nM T31391 CK0US2 122189874 IC50 = 980 nM T31391 C5V6NI 122189875 IC50 > 100000 nM T31391 CV7A9Y 122189876 IC50 > 100000 nM T31391 CN86VR 122189878 IC50 > 100000 nM T31391 C24OVE 122190735 IC50 = 1320 nM T31391 CSN6E0 122190738 IC50 = 24000 nM T31391 CD4EF9 122190739 IC50 = 1060 nM T31391 CVU5G7 122190835 IC50 = 2230 nM T31391 CB5X2Q 122190838 IC50 = 100000 nM T31391 CG69FQ 122190841 IC50 = 1250 nM T31391 CJ7X2U 122194794 IC50 = 1.5 nM T31391 C8XVB4 122194795 IC50 = 290 nM T31391 CL43TO 122194796 IC50 = 0.8 nM T31391 CAPX63 126456388 IC50 = 2.06 nM T31391 C0DUI4 126842756 IC50 = 1.33 nM T31391 CZXV13 126842761 IC50 = 0.76 nM T31391 CF7KI9 126842762 IC50 = 1.62 nM T31391 CG93JS 126842771 IC50 = 1.22 nM T31391 C6PLX9 127035081 IC50 = 4.9 nM T31391 CJ0KS7 127035239 IC50 = 2.3 nM T31391 CKSZ13 127035240 IC50 = 1.8 nM T31391 C6T1IM 127035241 IC50 = 5.7 nM T31391 CJRL72 127035242 IC50 = 0.7 nM T31391 CVKI59 127035243 IC50 = 1.9 nM T31391 CWJX95 127035244 IC50 = 2.3 nM T31391 C0XMS7 127035375 IC50 = 1.9 nM T31391 CMK5Q9 127035376 IC50 = 1.4 nM T31391 C4N7QB 127035377 IC50 = 1.6 nM T31391 CGN49F 127035378 IC50 = 4.3 nM T31391 C36UHW 127035569 IC50 = 0.3 nM T31391 CTKS36 127035740 IC50 = 3.7 nM T31391 CAXT02 127035741 IC50 = 3.2 nM T31391 CZB0L6 127035742 IC50 = 1.1 nM T31391 C4QWL5 127035743 IC50 = 1.3 nM T31391 CPGF39 127035744 IC50 = 1.8 nM T31391 CXTD34 127035745 IC50 = 1.8 nM T31391 CM98XR 127035752 IC50 = 1.7 nM T31391 C87MVA 127035753 IC50 = 1.7 nM T31391 CDW25O 127035754 IC50 = 0.4 nM T31391 CN08IS 127045827 IC50 > 100000 nM T31391 CAK85G 127046590 IC50 > 50000 nM T31391 CP3U8J 127046622 IC50 > 100000 nM T31391 CFAI71 127046624 IC50 = 56000 nM T31391 CB6PA7 127046626 IC50 > 100000 nM T31391 C76IGF 127046628 IC50 > 100000 nM T31391 CHL49F 127046630 IC50 = 790 nM T31391 CH0D2Z 127046632 IC50 = 4000 nM T31391 CK4SO7 127047730 IC50 = 2600 nM T31391 CSO9L3 127047731 IC50 = 19400 nM T31391 C4KIA9 127047732 IC50 = 16200 nM T31391 CHX41E 127047733 IC50 = 680 nM T31391 C6I7HW 127047734 IC50 = 34000 nM T31391 C2CP4F 127047761 IC50 > 100000 nM T31391 CYR1X2 127047762 IC50 > 100000 nM T31391 CIV4C2 127047839 IC50 > 100000 nM T31391 CDYA70 127047985 IC50 > 100000 nM T31391 C0FS5E 127048116 IC50 > 100000 nM T31391 C6NIM5 127048874 IC50 = 8.6 nM T31391 CXD69M 127048875 IC50 = 289 nM T31391 C65MAC 127048876 IC50 = 44 nM T31391 C23BWQ 127049179 IC50 = 1.4 nM T31391 CNCB06 127049180 IC50 = 1.9 nM T31391 CJ8SG3 127049204 IC50 = 1.5 nM T31391 CRM04V 127049507 IC50 = 0.5 nM T31391 C76VPA 127049823 IC50 = 54 nM T31391 CH0X6Q 127050132 IC50 = 0.5 nM T31391 CIGA32 127050759 IC50 = 1.1 nM T31391 CNY90B 127050760 IC50 = 1.5 nM T31391 C80WCY 127050761 IC50 = 0.6 nM T31391 CUVQ34 127050762 IC50 = 2.9 nM T31391 CJMS57 127051032 IC50 = 1.1 nM T31391 C9V4EG 127051045 IC50 = 0.7 nM T31391 C7W8JR 127051639 IC50 = 699 nM T31391 C36SXH 127052286 IC50 = 1.1 nM T31391 CBR1F8 127052287 IC50 = 26 nM T31391 CHZX75 127052288 IC50 = 0.6 nM T31391 CB34GQ 127052289 IC50 = 0.7 nM T31391 CLG0Q3 127052290 IC50 = 16 nM T31391 CL2S0F 127052581 IC50 = 1.7 nM T31391 C1W5AL 127052582 IC50 = 155 nM T31391 C4TI8H 127052590 IC50 = 1170 nM T31391 CNV0A8 127052636 IC50 = 0.56 nM T31391 CS2Z9R 127052637 IC50 = 0.23 nM T31391 C75EAL 127052638 IC50 = 0.24 nM T31391 CRP1K2 130385241 IC50 = 5.8 nM T31391 CTIO26 130385242 IC50 = 5.17 nM T31391 C30ERZ 130385243 IC50 = 1.9 nM T31391 C09MJL 130385246 IC50 = 205.2 nM T31391 CZ29WO 130385251 IC50 = 19.64 nM T31391 CED01R 130385253 IC50 = 14.95 nM T31391 C83CDX 130385258 IC50 = 8.42 nM T31391 CB37AX 130385267 IC50 = 216.2 nM T31391 C5DWM6 130391940 IC50 = 70.42 nM T31391 C41QVU 130391961 IC50 = 6.13 nM T31391 C6PMX7 130391978 IC50 = 17.65 nM T31391 CD7B2H 130392003 IC50 = 8.91 nM T31391 C15BEV 130392042 IC50 = 563.9 nM T31391 CD6C4U 130392043 IC50 = 13070 nM T31391 CH9E4W 132055397 IC50 = 110.1 nM T31391 C6CV5J 132069286 IC50 = 154.67 nM T31391 CALB73 134131859 IC50 = 5400 nM T31391 CA5Y0V 134132454 IC50 = 250 nM T31391 CMY0V5 134132485 IC50 = 5000 nM T31391 CTZU69 134132901 IC50 = 14.6 nM T31391 CH1G3A 134133219 IC50 = 260 nM T31391 CS9K7A 134133834 IC50 = 360 nM T31391 C2BA5L 134134276 IC50 = 890 nM T31391 CVE96U 134134571 IC50 = 300 nM T31391 CB59UX 134135207 IC50 = 73 nM T31391 CIXJ53 134135875 IC50 = 250 nM T31391 C4Q2GB 134136466 IC50 = 121.56 nM T31391 C5OS4T 134136634 IC50 = 39.2 nM T31391 C14XET 134137196 IC50 = 140 nM T31391 CMB8T7 134137851 IC50 = 32.64 nM T31391 CTP9X4 134138048 IC50 = 21520 nM T31391 C58KIQ 134138807 IC50 = 500 nM T31391 C2OWQ1 134138838 IC50 = 760 nM T31391 CPLI26 134139792 IC50 = 400 nM T31391 CDV6U9 134140856 IC50 = 49.73 nM T31391 C5TS2J 134141415 IC50 = 2600 nM T31391 CB8QD9 134142015 IC50 = 770 nM T31391 CY2CJ4 134142362 IC50 = 510 nM T31391 CK27IY 134143858 IC50 = 2930 nM T31391 CKP0Z5 134144315 IC50 = 78.33 nM T31391 COT7P4 134144691 IC50 = 206.71 nM T31391 CD0XT6 134145610 IC50 = 800 nM T31391 C8B3CU 134150931 IC50 = 280 nM T31391 CEC9Y2 134151020 IC50 = 50860 nM T31391 C0G5PV 134151859 IC50 = 220 nM T31391 C3NF8J 134151937 IC50 = 140 nM T31391 CQRM94 134152842 IC50 = 360 nM T31391 C6TL9Z 134153173 IC50 = 950 nM T31391 CBN6Z7 134153444 IC50 = 610 nM T31391 CZX9V0 134154214 IC50 = 337.8 nM T31391 C4ZWS1 134157002 IC50 = 120 nM T31391 CNO0R1 135411740 IC50 = 2120 nM T31391 CRM4Q8 135518358 IC50 = 3 nM T31391 CMI5A6 135964368 IC50 = 95 nM T31391 CC4L2F 136060652 IC50 > 3000 nM T31391 CP7BS2 136098501 IC50 = 6113 nM T31391 CO04QA 136177302 IC50 = 7 nM T31391 C1GYM8 136411530 IC50 = 11 nM T31391 CR4VI2 137225025 IC50 = 0.6 nM T31391 CAN18C 137631813 IC50 = 2.1 nM T31391 C95BML 137632265 IC50 = 70 nM T31391 C5H2EA 137637131 IC50 = 27.54 nM T31391 C2FA1T 137637208 IC50 = 7.2 nM T31391 CS2L6B 137637588 IC50 = 43.4 nM T31391 CO9BH6 137638100 IC50 = 50.2 nM T31391 C6IJ3A 137642352 IC50 = 8.5 nM T31391 CY0R4C 137644720 IC50 = 60 nM T31391 CI8FG2 137644837 IC50 = 1200 nM T31391 C1MBC4 137646578 IC50 = 31.8 nM T31391 C67NZA 137650009 IC50 = 123.3 nM T31391 C8BH1R 137650030 IC50 = 537 nM T31391 CG8HS3 137652269 IC50 = 29 nM T31391 C9SX0Q 137653253 IC50 = 139 nM T31391 CH4MT1 137655300 IC50 = 8.7 nM T31391 CV5A3F 137657117 IC50 = 470 nM T31391 CKF03W 137659671 IC50 = 5.5 nM T31391 C2MV9K 137661375 IC50 = 151.7 nM T31391 CJT56Y 137662038 IC50 = 2.6 nM T31391 CO6JA3 141514759 IC50 = 188.7 nM T31391 C1SQ2R 141514762 IC50 = 64.47 nM T31391 CHI84B 141514764 IC50 = 65.36 nM T31391 C3SKH4 145948172 IC50 = 97 nM T31391 C8S7FY 145949528 IC50 = 1.45 nM T31391 CR2UP9 145950777 IC50 > 100 nM T31391 C7IZU2 145950786 IC50 = 1.61 nM T31391 C7SMW4 145951086 IC50 = 0.72 nM T31391 CR5AJ7 145952072 IC50 = 26.6 nM T31391 C2MWR4 145952134 IC50 = 15.3 nM T31391 CV30OD 145952476 IC50 = 0.77 nM T31391 CBFR49 145953292 IC50 = 1.69 nM T31391 CYF24S 145953544 IC50 = 0.76 nM T31391 C38IOE 145953726 IC50 = 0.61 nM T31391 C4JQT5 145953757 IC50 > 100 nM T31391 C0C4KJ 145954860 IC50 = 0.79 nM T31391 C48AXH 145955793 IC50 = 2.4 nM T31391 C6QY1K 145957483 IC50 = 1.58 nM T31391 CMO0J1 145957949 IC50 = 1.67 nM T31391 C35FNU 145957994 IC50 = 18 nM T31391 CR9S6F 145958227 IC50 = 2.3 nM T31391 CB72HG 145958828 IC50 = 1.25 nM T31391 C60WXK 145959997 IC50 = 0.77 nM T31391 C8V5PA 145962482 IC50 = 0.54 nM T31391 CBL76R 145964231 IC50 = 2500 nM T31391 CF53NA 145964407 IC50 = 400 nM T31391 CNMT16 145965136 IC50 = 1200 nM T31391 CQW63D 145965301 IC50 = 11500 nM T31391 C6D0VY 145967130 IC50 = 21500 nM T31391 CI82EJ 145973071 IC50 = 10400 nM T31391 C1Y5FP 145973406 IC50 = 6.8 nM T31391 CP8EN1 145973616 IC50 = 0.54 nM T31391 CP7VT2 145973710 IC50 = 1300 nM T31391 C2C1ZR 145974002 IC50 = 17200 nM T31391 C9C4WU 145975568 IC50 = 80 nM T31391 CRNK53 145977284 IC50 = 46500 nM T31391 CWF4Y7 145977953 IC50 = 2000 nM T31391 CB3K0Q 145978529 IC50 = 59900 nM T31391 CR3I9D 145978547 IC50 = 49 nM T31391 CNG4Z2 145983347 IC50 = 1.12 nM T31391 CH6P8Q 145983352 IC50 = 1270 nM T31391 C02BLT 145983464 IC50 = 7580 nM T31391 CN1V6D 145984069 IC50 = 28050 nM T31391 C3QT0G 145984247 IC50 = 1780 nM T31391 CMWH26 145984429 IC50 = 15780 nM T31391 CL6D3F 145984547 IC50 = 19.6 nM T31391 CIX4P5 145985997 IC50 = 232.8 nM T31391 CM6L4K 155510749 IC50 = 190 nM T31391 C5ZQ7W 155511281 IC50 = 2.91 nM T31391 CP4SH8 155511399 IC50 > 100000 nM T31391 CEL39X 155511987 IC50 = 74.6 nM T31391 CQA73O 155512586 IC50 = 197 nM T31391 C57QZJ 155512836 IC50 = 7.6 nM T31391 CX3U8Z 155515016 IC50 = 10.21 nM T31391 C7FOS5 155516136 IC50 = 538 nM T31391 CTE94M 155516800 IC50 > 10000 nM T31391 C19ZCJ 155518265 IC50 = 395 nM T31391 C8UOJ4 155518381 IC50 = 1.7 nM T31391 C8U9ON 155518908 Ki = 217.9 nM T31391 CW0NI8 155519444 IC50 = 0.1 nM T31391 C7O2UF 155519988 IC50 > 100000 nM T31391 C3I8AW 155520161 IC50 = 60 nM T31391 C1Z2NP 155522069 Ki = 152.8 nM T31391 C4AZ9V 155523785 IC50 = 93.2 nM T31391 CG18KV 155524302 IC50 = 0.75 nM T31391 C0RAC6 155524362 IC50 = 3900 nM T31391 CTSA30 155526359 IC50 = 5.61 nM T31391 CVD89H 155526728 IC50 = 208 nM T31391 C5C4UV 155526759 IC50 = 5.99 nM T31391 CAT3J0 155526949 IC50 = 3.9 nM T31391 C7J4VQ 155527859 IC50 = 1.75 nM T31391 CLE9I0 155528648 IC50 = 0.22 nM T31391 C3LT9C 155529752 IC50 > 100000 nM T31391 C8FHJ2 155529886 IC50 = 2.43 nM T31391 CCX9H6 155530472 IC50 = 226 nM T31391 C7YP3B 155530585 IC50 = 4.41 nM T31391 C2YWG1 155530817 IC50 = 790 nM T31391 CB6N4S 155531120 IC50 = 0.18 nM T31391 CGV6C1 155531169 IC50 = 22.09 nM T31391 CEOQ32 155531330 IC50 = 50.9 nM T31391 CMY59I 155531892 IC50 > 100000 nM T31391 C0ZCE3 155533243 IC50 = 89.8 nM T31391 CN04KW 155533304 IC50 = 74.43 nM T31391 C95ZUT 155534726 Ki = 180.8 nM T31391 CW8Z1X 155535213 IC50 > 100000 nM T31391 CA9Z6Q 155538747 IC50 = 121300 nM T31391 CG3RS6 155540249 IC50 = 223 nM T31391 CJ67GL 155540375 IC50 = 3.5 nM T31391 CM1FA9 155544265 Ki = 380.1 nM T31391 CY25EZ 155544299 IC50 = 4.6 nM T31391 C8H3MJ 155544665 IC50 = 20.48 nM T31391 CU17DA 155544967 IC50 = 2.35 nM T31391 CY2V6P 155545256 IC50 = 2.25 nM T31391 C62YMT 155545522 IC50 = 85.48 nM T31391 CMS63L 155545906 IC50 = 56.6 nM T31391 CGZ08R 155547532 IC50 = 3830000 nM T31391 CDGW26 155547608 IC50 = 76170 nM T31391 CNA9X4 155548276 IC50 = 217 nM T31391 CWF0L6 155548277 IC50 = 483 nM T31391 CM9K4B 155548792 IC50 = 0.72 nM T31391 CB1AF4 155549522 IC50 = 7.5 nM T31391 CL9R1Y 155549582 IC50 > 100000 nM T31391 C3MW1B 155550953 IC50 > 10000 nM T31391 CX9Y4B 155552378 IC50 = 1.05 nM T31391 C8XSI3 155553379 IC50 = 2 nM T31391 C6QKL9 155553392 Ki = 412.2 nM T31391 C1D5QZ 155554658 IC50 = 2.5 nM T31391 CR8AU9 155555628 IC50 = 68510 nM T31391 C1GD0E 155555672 Ki = 941.2 nM T31391 CHV85S 155556058 IC50 > 100000 nM T31391 C6N4WH 155557237 IC50 > 100000 nM T31391 CSCD34 155559193 IC50 > 100000 nM T31391 C7KVR5 155559306 IC50 = 3.9 nM T31391 CRL47X 155559391 IC50 = 28.7 nM T31391 C1NE4T 155560255 IC50 > 100000 nM T31391 C68CRH 155561682 IC50 = 4 nM T31391 CQ7JL5 155562412 IC50 = 55870 nM T31391 C90QLF 155563643 Ki = 103.7 nM T31391 C48ETF 155565121 IC50 = 170 nM T31391 CUL27B 155565517 Ki = 341.6 nM T31391 CE5SI7 155566076 IC50 > 100000 nM T31391 CI5C6P 155568161 IC50 = 0.44 nM T31391 CUQL05 155568269 IC50 = 5.06 nM T31391 CDB0S2 155568427 IC50 = 421 nM T31391 D00HSG 44408767 IC50 = 3300 nM T31391 D00KMP 44431763 IC50 = 5300 nM T31391 D00RIX 5280443 IC50 = 140 nM T31391 D00YEV 5281605 IC50 > 200000 nM T31391 D02RDY 11375559 IC50 > 100000 nM T31391 D02RIE 44440628 Ki = 13000 nM T31391 D02WBC 3847395 IC50 = 33000 nM T31391 D03DNV 71655266 IC50 > 100000 nM T31391 D04CAR 10607286 Ki = 0.4 nM T31391 D05LYC 11403745 IC50 = 140 nM T31391 D05UUA 16049437 Ki = 820 nM T31391 D05XWX 10130510 Ki = 3.8 nM T31391 D06AUB 44440618 Ki = 3400 nM T31391 D06NRU 1393052 IC50 = 2300 nM T31391 D06UKY 44440632 Ki = 2800 nM T31391 D07ALM 11232124 Ki = 0.082 nM T31391 D07HWI 6931234 IC50 = 75000 nM T31391 D07IJU 13578534 Ki = 2100 nM T31391 D08NMS 46900258 Ki = 1.4 nM T31391 D09ALJ 5280805 IC50 = 145000 nM T31391 D09BYA 44431745 IC50 = 3500 nM T31391 D09MVE 263366 IC50 = 30000 nM T31391 D0AU0M 637542 IC50 = 83180 nM T31391 D0CP1J 56658139 IC50 > 50000 nM T31391 D0G3TK 5280863 IC50 = 132000 nM T31391 D0JI3S 11674875 IC50 = 18600 nM T31391 D0JL2T 5393152 IC50 > 200000 nM T31391 D0L5RI 44328273 Ki = 7880 nM T31391 D0L9XR 447256 Ki = 470 nM T31391 D0N1FU 6918465 Ki = 126 nM T31391 D0N1QQ 94701 Ki = 2200 nM T31391 D0N5CI 11615508 IC50 = 12000 nM T31391 D0O9RD 44403067 Ki = 3350 nM T31391 D0P5OE 2724998 IC50 = 45000 nM T31391 D0PB2M 23645372 Ki = 34 nM T31391 D0R5OE 44422449 IC50 = 538 nM T31391 D0S0RK 10680 IC50 = 170 nM T31391 D0T2EW 11075394 Ki = 1.4 nM T31391 D0T3PW 5281672 IC50 = 37150 nM T31391 D0U4HG 23634523 IC50 > 36900 nM T31391 D0V9EN 689043 IC50 = 3370 nM T31391 D0W4GM 205131 IC50 = 40000 nM T31391 D0X0IF 23655936 IC50 > 39100 nM T31391 D0X2JG 2777206 IC50 = 37000 nM T31391 D0Y3TZ 370 IC50 = 4650 nM T31391 D0Y5IQ 44255320 IC50 = 10000 nM T02439 CJ6R1L 18445508 IC50 = 199.53 nM T02439 C3HVM7 18445520 IC50 = 31.62 nM T02439 C8OR0L 18445737 IC50 = 3162.28 nM T02439 CM28GF 18445739 IC50 = 63.1 nM T02439 C0TC2X 18445833 IC50 = 630.96 nM T02439 C3VRO9 44557921 IC50 > 10000 nM T02439 CL0OC7 45375855 IC50 = 2511.89 nM T02439 CZXJ98 45483394 IC50 = 125.89 nM T02439 C25NVM 45483417 IC50 = 316.23 nM T02439 C0I2MB 45483418 IC50 = 251.19 nM T02439 C6CJ2N 45483436 IC50 = 794.33 nM T02439 CZOK17 45483447 IC50 = 1000 nM T02439 C1W0AX 45483460 IC50 = 1000 nM T02439 CICD40 45483461 IC50 = 2511.89 nM T02439 CXK2H9 45483468 IC50 = 1584.89 nM T02439 C7MQI8 45483469 IC50 > 10000 nM T02439 CED7U8 45483470 IC50 = 50.12 nM T02439 CBV30W 45483507 IC50 = 501.19 nM T02439 CAL8P6 45483508 IC50 = 794.33 nM T02439 C2UPW3 45483509 IC50 = 1258.93 nM T02439 CA23TC 45483510 IC50 = 7.943 nM T02439 CZC96T 45483513 IC50 = 19.95 nM T02439 C2ABD6 45483530 IC50 = 251.19 nM T02439 C4EZO3 45483716 IC50 = 63.1 nM T02439 CB3N6J 45483717 IC50 = 501.19 nM T02439 CH1S9G 45483725 IC50 = 79.43 nM T02439 CE6K8L 45483734 IC50 > 10000 nM T02439 C4DG0Z 45483735 IC50 > 10000 nM T02439 CXB94H 53466728 IC50 = 17020 nM T02439 CYQ41S 53466951 IC50 = 1863 nM T02439 CX0R1K 53469059 IC50 = 460 nM T02439 CV7C0D 53469060 IC50 = 37 nM T02439 CCKD45 53469061 IC50 = 61 nM T02439 C91STB 53469449 IC50 = 214 nM T02439 CZ1CI3 53469824 IC50 = 12080 nM T02439 CX4H6I 86583042 IC50 > 10000 nM T02439 C4TXF2 118730409 IC50 > 10000 nM T02439 CXC69T 137321158 IC50 = 26 nM T02439 C2MD1Q 155513187 IC50 > 10000 nM T02439 D02LIR 45375987 IC50 = 6.31 nM T02439 D0N4LR 53469448 IC50 = 420 nM T15023 C31FHD 156080 IC50 = 25000 nM T15023 CC7OA9 9854089 IC50 = 84100 nM T15023 CHKV76 15984054 IC50 = 2000 nM T15023 C0VBC2 22779253 IC50 = 9300 nM T15023 COB8R4 24765913 IC50 = 13000 nM T15023 CS5O8W 24815567 IC50 = 14000 nM T15023 C6UM9C 24815571 IC50 = 52000 nM T15023 CX0BK1 24815653 IC50 = 18000 nM T15023 CCPS98 24815654 IC50 = 9000 nM T15023 C3V9CG 24815655 IC50 = 17000 nM T15023 CT86UJ 24815656 IC50 = 33000 nM T15023 CPZQ89 44415045 IC50 = 80000 nM T15023 CI8GD1 44415050 IC50 = 3000 nM T15023 CFK0E3 44415051 IC50 = 3000 nM T15023 CJ5O9B 44415067 IC50 = 62000 nM T15023 CGIB09 44415068 IC50 = 60000 nM T15023 CQ0P6M 44415069 IC50 = 3000 nM T15023 CJ51WK 44415070 IC50 = 3000 nM T15023 C09FPC 44415084 IC50 = 47000 nM T15023 C2X0IH 44415085 IC50 = 43000 nM T15023 CUK58S 44415107 IC50 = 19000 nM T15023 CCO95R 44415108 IC50 = 13000 nM T15023 CALV50 44415122 IC50 = 9000 nM T15023 C8DT5W 44415123 IC50 = 4000 nM T15023 C8DA3X 44415134 IC50 = 4000 nM T15023 C4E6OP 44415135 IC50 = 3000 nM T15023 C7K9YM 44415146 IC50 = 2000 nM T15023 C4CRI6 44415160 IC50 = 95000 nM T15023 C7H6QP 44415168 IC50 = 22000 nM T15023 C95GPD 44415171 IC50 = 14000 nM T15023 CXUY04 44415198 IC50 = 13000 nM T15023 C7MAV1 44415199 IC50 = 13000 nM T15023 CD3X5N 44415203 IC50 = 10000 nM T15023 CQ4Y6E 44415204 IC50 = 10000 nM T15023 CUBP89 44415228 IC50 = 29000 nM T15023 C2FL1O 44415229 IC50 = 9000 nM T15023 CEJH97 44415230 IC50 = 6000 nM T15023 CSGQ74 44415243 IC50 = 6000 nM T15023 CN5F8H 44415244 IC50 = 6000 nM T15023 C3RB4Q 44415264 IC50 = 5000 nM T15023 CGU69B 44415265 IC50 = 5000 nM T15023 CWJ86B 44415284 IC50 = 79000 nM T15023 CG4O3L 44415285 IC50 = 42000 nM T15023 C1TGL7 44415286 IC50 = 5000 nM T15023 C5QZO0 44415287 IC50 = 4000 nM T15023 C7PXM4 44415303 IC50 = 4000 nM T15023 CL5SJ9 44415321 IC50 = 3000 nM T15023 CW2V1K 44415322 IC50 = 2000 nM T15023 CF2B9J 44415323 IC50 = 2000 nM T15023 CMXN47 44415328 IC50 = 2000 nM T15023 C4CO0Q 44415329 IC50 = 2000 nM T15023 CXNB21 44631827 IC50 = 3000 nM T15023 CFS01Z 45139618 IC50 = 17000 nM T15023 C3FIO4 45139619 IC50 = 12000 nM T15023 CYV65U 45139620 IC50 = 6000 nM T15023 C6F4MD 46881769 IC50 = 30000 nM T15023 CD53IC 46888232 IC50 = 92000 nM T15023 CSZN86 73345690 IC50 = 18000 nM T15023 C1V4YX 117919744 IC50 = 8900 nM T15023 CN3XO8 133081972 IC50 = 1600 nM T15023 CH63VL 145979165 IC50 = 800 nM T15023 CLP5J8 155510478 IC50 = 10715.19 nM T15023 C8BHO5 155519379 IC50 = 120000 nM T15023 CM7XI4 155521636 IC50 = 26000 nM T15023 C89PUV 155535868 IC50 = 187000 nM T15023 C62ATN 155538638 IC50 = 2951.21 nM T15023 CC39XR 155539536 IC50 = 50100 nM T15023 CV7JH9 155541491 IC50 = 20900 nM T15023 CKF02B 155541869 IC50 = 181000 nM T15023 CDP3A5 155542006 IC50 = 2884.03 nM T15023 C4LT0D 155542021 IC50 = 16000 nM T15023 CKR03L 155542693 IC50 = 18100 nM T15023 CUX2Z1 155543565 IC50 = 7700 nM T15023 CN2GQ1 155544385 IC50 = 16100 nM T15023 CF79TY 155545026 IC50 = 23400 nM T15023 CRA0T4 155545299 IC50 = 15848.93 nM T15023 C6TJV0 155545675 IC50 = 9200 nM T15023 C3U9ID 155545743 IC50 = 2300 nM T15023 C5C0LF 155548104 IC50 = 21300 nM T15023 CUS5A3 155549314 IC50 = 88000 nM T15023 CZGJ90 155549636 IC50 = 39000 nM T15023 C73BNV 155550340 IC50 > 100000 nM T15023 C06ERO 155552650 IC50 = 48600 nM T15023 CY9T5X 155554019 IC50 = 69000 nM T15023 CVIM57 155555240 IC50 = 14000 nM T15023 C2ROS0 155556517 IC50 = 80500 nM T15023 C2HMC4 155557562 IC50 = 21300 nM T15023 C84LDU 155560254 IC50 > 100000 nM T15023 CP6GZ9 155560763 IC50 = 134000 nM T15023 CCN1U7 155566104 IC50 = 21300 nM T15023 CQ4E5Y 155566947 IC50 = 5370.32 nM T15023 CBE1X8 155569690 IC50 = 7200 nM T15023 D0GD5G 15858500 IC50 = 4600 nM T00563 D09JEJ 24748573 IC50 = 11 nM T00563 D0E3TC 44259 IC50 = 844 nM T00563 D02GEJ 5326976 Ki = 112 nM T00563 CJH12X 537952 IC50 = 32200 nM T00563 CR9EJ0 11352337 Ki = 35 nM T00563 C8V7ZF 11352967 Ki = 37 nM T00563 CV78IN 16224258 IC50 = 190 nM T00563 CY8X0J 24811794 IC50 = 701 nM T00563 C4HY6I 44263430 Ki = 21 nM T00563 CYX19V 44263445 Ki = 78 nM T00563 C0RK5W 44263447 Ki = 62 nM T00563 CNZ19H 44263451 Ki = 342 nM T00563 C3VRO9 44557921 IC50 > 10000 nM T00563 CDK93W 56946894 IC50 < 3000 nM T00563 CE2DU7 56968171 Ki = 188 nM T00563 C4RIA1 56968172 Ki = 93 nM T00563 CYIO69 56968174 Ki = 31 nM T00563 CT1ZJ3 56968175 Ki = 55 nM T00563 C73NVJ 56968176 Ki = 44 nM T00563 C0MS9N 56968177 Ki = 83 nM T00563 C8WDK1 57342036 IC50 = 11 nM T00563 C0I6SZ 57342039 IC50 = 32000 nM T00563 CA7BS4 57342210 IC50 = 63 nM T00563 CVBF89 57342215 IC50 = 25000 nM T00563 C8P1ZB 57342375 IC50 = 5300 nM T00563 CH6RV3 57342376 IC50 = 3300 nM T00563 C65NOS 57342377 IC50 = 1700 nM T00563 C8TFC7 57342378 IC50 = 1200 nM T00563 CZ0R4K 57342379 IC50 = 5800 nM T00563 C8U4MB 57342380 IC50 = 1800 nM T00563 CJSO14 57342381 IC50 = 2800 nM T00563 CW3P9K 57342382 IC50 = 4300 nM T00563 CFX60S 57342541 IC50 = 1600 nM T00563 CF9BZ1 57342542 IC50 = 2900 nM T00563 C2C4XB 57342543 IC50 = 4300 nM T00563 C9XPF2 57342544 IC50 = 2700 nM T00563 C9MA4U 57342545 IC50 = 3000 nM T00563 CWZY51 57342546 IC50 = 8200 nM T00563 CK9IC1 57342547 IC50 = 3100 nM T00563 CO14NX 57342548 IC50 = 5700 nM T00563 CTNX36 57342718 IC50 = 2400 nM T00563 C8G6RK 57342719 IC50 = 2100 nM T00563 CJ9OF3 57400663 Ki = 24 nM T00563 CV63UL 67240318 IC50 > 10000 nM T00563 CDE3Y9 76321032 IC50 < 4000 nM T00563 C4T7YB 127025199 IC50 = 4.6 nM T00563 CP02TW 127025200 IC50 = 10 nM T00563 C57ECS 127025201 IC50 = 280 nM T00563 CP31UE 127025202 IC50 = 10 nM T00563 CHP6R9 127025499 IC50 = 12 nM T00563 CY37QE 127025500 IC50 = 12 nM T00563 CR59LY 127026094 IC50 = 11 nM T00563 CWIG59 127026095 IC50 = 9.8 nM T00563 C45BZG 127026096 IC50 = 160 nM T00563 C0HLT9 127026097 IC50 = 19 nM T00563 CW5JB1 127026098 IC50 = 14 nM T00563 CL4CG5 127026727 IC50 = 13 nM T00563 CO6X5B 127026728 IC50 = 11 nM T00563 CA5XG8 127026729 IC50 = 9.5 nM T00563 C6EIR3 127027657 IC50 = 9.6 nM T00563 C1MF5T 127029513 IC50 = 8.8 nM T00563 C86HPW 155518524 IC50 = 99000 nM T00563 D0CP3M 5149739 Ki = 270 nM T00563 D0K6BI 46943415 Ki = 21 nM T00563 D0US9O 45275255 IC50 = 2.7 nM T44351 D0P1FO 16078 Ki = 41 nM T44351 D0YZ8I 4273754 Ki = 164 nM T44351 D0J7RW 5311501 Ki = 24 nM T44351 CRM5P4 9845561 Ki = 0.46 nM T44351 C7SW3C 10360860 Ki = 9.5 nM T44351 C2FK8Z 13645595 Ki > 10000 nM T44351 C52FSE 24096428 Ki = 0.77 nM T44351 C3MZ0J 44327221 Ki = 0.81 nM T44351 CIBP20 44327403 Ki = 0.6 nM T44351 CX03ZD 44327404 Ki = 0.84 nM T44351 CG59OH 44327429 Ki = 0.46 nM T44351 CLH31M 44368310 Ki = 22 nM T44351 C52UYW 44368361 Ki = 1250 nM T44351 CETG63 44368362 Ki = 46 nM T44351 CIZ10X 44368367 Ki > 10000 nM T44351 CG92UC 44368388 Ki = 48 nM T44351 CLK34Y 44368424 Ki = 81 nM T44351 C52RNY 44368441 Ki = 72 nM T44351 CTKI30 44368442 Ki = 33 nM T44351 C83XUB 44368703 Ki > 10000 nM T44351 CO0RU5 44371487 Ki = 800 nM T44351 CY92LZ 53310757 Ki > 1000 nM T44351 D04GDY 638026 Ki = 44 nM T44351 D0D6OH 104895 Ki = 0.924 nM T44351 D0F4BX 9821569 Ki = 0.73 nM T01138 D01GBY 124087 IC50 = 172000 nM T01138 D06ABF 3957 IC50 = 4000 nM T01138 D0S1CQ 133017 IC50 > 40000 nM T01138 D0C2HI 60680 IC50 = 54800 nM T01138 C0TSD5 31843 IC50 > 80000 nM T01138 CA95CK 4161540 IC50 = 18300 nM T01138 CL4VY5 10137458 IC50 = 16100 nM T01138 CQWE69 10363386 IC50 = 4600 nM T01138 CF97IO 14554122 IC50 = 26400 nM T01138 CZQM08 14554127 IC50 = 4900 nM T01138 CSXR86 14554128 IC50 = 5300 nM T01138 CJU02M 14554129 IC50 = 36000 nM T01138 C80GMR 18337326 IC50 > 80000 nM T01138 C8RD9C 18337327 IC50 > 80000 nM T01138 CI2W9S 18337331 IC50 = 7800 nM T01138 C71YDN 18337336 IC50 = 19600 nM T01138 C9RWZ3 18382725 IC50 = 4500 nM T01138 C74WSR 20659961 IC50 = 5700 nM T01138 COP68C 22914796 IC50 = 22900 nM T01138 C29SNE 29918864 IC50 = 17600 nM T01138 CFGH46 29976517 IC50 > 80000 nM T01138 C5F8WR 29976521 IC50 > 80000 nM T01138 C5GW8F 29981724 IC50 > 80000 nM T01138 C9MZ5R 29983056 IC50 = 12400 nM T01138 CLK4Y7 59047051 IC50 = 14800 nM T01138 CS2N1P 118721922 IC50 = 35000 nM T01138 C5CV9A 118721923 IC50 > 80000 nM T01138 CB3L9V 118721924 IC50 = 16800 nM T01138 CGE6B0 118721925 IC50 > 80000 nM T01138 CZF1A9 118721926 IC50 = 4900 nM T01138 CVI2B6 118721927 IC50 = 41500 nM T01138 C2K6ML 118721928 IC50 = 5000 nM T01138 C6YF0A 118721929 IC50 = 10800 nM T01138 CK03VE 118721930 IC50 = 3400 nM T01138 CD0O2N 118721931 IC50 = 5200 nM T01138 C7JP0Z 118721932 IC50 = 18700 nM T01138 CI56NQ 118721933 IC50 = 39100 nM T01138 CBM7V0 118721934 IC50 = 7700 nM T03634 D07SDQ 969516 IC50 = 25000 nM T03634 D0PH9I 118693659 Ki = 6309.57 nM T03634 D0U2BH 65064 IC50 = 50000 nM T03634 D0ZW4W 46907787 IC50 = 9600 nM T03634 CZI4N9 13387 IC50 = 2300000 nM T03634 C5XSG3 19868 IC50 = 32000 nM T03634 C76RDA 43000 IC50 > 50000 nM T03634 CFAL50 43001 IC50 > 50000 nM T03634 CZX1K3 223771 IC50 > 200000 nM T03634 CJ6X2Y 572983 IC50 = 10000 nM T03634 CAT79Z 589098 IC50 = 99000 nM T03634 CG5O0H 638578 IC50 = 11800 nM T03634 CM1EX8 735746 IC50 > 2000000 nM T03634 COP70H 735747 IC50 = 27000 nM T03634 CGR7Y5 755980 IC50 > 50000 nM T03634 CBG2A0 1078352 IC50 = 230 nM T03634 CVF47X 1238761 IC50 > 50000 nM T03634 CML94F 1415890 IC50 = 30000 nM T03634 C2M0SE 1511198 IC50 = 1584.89 nM T03634 CJK1F0 1511199 IC50 = 1258.93 nM T03634 CJWR09 1561807 IC50 = 41000 nM T03634 CS05BM 1600566 IC50 = 115700 nM T03634 C6XQA3 1797300 IC50 = 3200 nM T03634 CE17KZ 1821586 IC50 = 9110 nM T03634 CH01FB 2054569 IC50 = 41360 nM T03634 COZK67 2728636 IC50 = 7000 nM T03634 CV8A1O 2763642 IC50 = 1900000 nM T03634 C3GU6L 2766364 IC50 = 40000 nM T03634 CXD3U8 3152392 IC50 > 200000 nM T03634 C9GO8K 3326945 IC50 > 50000 nM T03634 C2P6IC 3846558 IC50 = 29400 nM T03634 CJ73FZ 4247469 IC50 = 440 nM T03634 CR3SF5 4907545 IC50 = 15848.93 nM T03634 CWG19Q 4908238 IC50 = 6309.57 nM T03634 CUGH30 5157255 IC50 > 50000 nM T03634 CO1H6V 5304236 IC50 = 1440 nM T03634 C8BZ9Y 5325760 IC50 > 200000 nM T03634 CQCH54 6210261 IC50 = 60000 nM T03634 CV67KR 6490661 IC50 = 16730 nM T03634 CH41UK 9992116 IC50 = 2500 nM T03634 CV47EZ 10081070 IC50 = 500000 nM T03634 CUD8X4 10355367 IC50 = 5280 nM T03634 C93EDN 10442296 IC50 > 100000 nM T03634 CK8O6Q 11238147 IC50 = 3000 nM T03634 CT53WA 12206142 IC50 > 200000 nM T03634 C75UZW 12564532 IC50 = 455000 nM T03634 C34GWI 12622087 IC50 = 12000 nM T03634 CE24BV 12689741 IC50 > 50000 nM T03634 C7U9KW 13099766 IC50 = 1950 nM T03634 CCSB13 16662818 IC50 = 1670 nM T03634 C49GBY 27604952 IC50 = 3000 nM T03634 C3UFS6 39791103 IC50 = 3400 nM T03634 C1OEL5 40889550 IC50 = 23000 nM T03634 C2P0IW 44243549 IC50 = 55700 nM T03634 C8XFC2 45494549 IC50 = 13620 nM T03634 CEK9S5 45917950 IC50 > 50000 nM T03634 CV92LK 46786182 IC50 > 50000 nM T03634 CHFE80 51081283 IC50 > 100000 nM T03634 C35MQH 51371083 IC50 = 270 nM T03634 CFX06I 51721279 IC50 = 6800 nM T03634 CG3PR6 52912222 IC50 = 31622.78 nM T03634 C4XCJ0 53257845 IC50 = 2850 nM T03634 CQEF28 53308655 IC50 = 32200 nM T03634 CEK3X6 54757749 IC50 = 86900 nM T03634 C1D3WH 54757750 IC50 = 45400 nM T03634 C1DZ7Y 54757751 IC50 = 49400 nM T03634 C6W5OZ 54757752 IC50 = 12900 nM T03634 CBOE48 56669892 IC50 = 1270 nM T03634 CT76FH 56877138 IC50 = 55000 nM T03634 CCGW97 60149330 IC50 = 758 nM T03634 C6KWC8 69236418 IC50 = 130000 nM T03634 C9L0KD 70699440 IC50 = 1100 nM T03634 CV7OR2 70699441 IC50 = 771 nM T03634 C4MJ0T 71624784 IC50 = 4100 nM T03634 CIX91F 71624785 IC50 = 6300 nM T03634 C1D8GF 71624786 IC50 = 8600 nM T03634 C3R9WA 71624787 IC50 = 8500 nM T03634 CLQ1X8 71624896 IC50 = 10800 nM T03634 CODK30 71624901 IC50 = 3960 nM T03634 CI15JC 71624902 IC50 = 2070 nM T03634 CLZ7C8 71624903 IC50 = 2810 nM T03634 CIPN50 71760902 IC50 = 1000 nM T03634 CA81BL 72201025 IC50 = 240 nM T03634 CQ78NK 76310219 IC50 = 199.53 nM T03634 CM4J8Q 76317442 IC50 = 630.96 nM T03634 CM7TH3 76328466 IC50 = 794.33 nM T03634 C0T5NK 76335637 IC50 = 630.96 nM T03634 C5TB9S 77843982 IC50 = 1000 nM T03634 CL3R7M 81689862 IC50 = 1000 nM T03634 CB9AL4 86287631 IC50 = 3700 nM T03634 CYQ91J 90667397 IC50 = 3980 nM T03634 CS3W6O 90667751 IC50 = 40900 nM T03634 CZBD29 90667752 IC50 = 28400 nM T03634 CF4W8Q 90667754 IC50 = 35900 nM T03634 C2B4NA 90667755 IC50 = 38500 nM T03634 C32KSA 91808023 IC50 = 8700 nM T03634 CTA46H 91826273 IC50 = 1100 nM T03634 C0N1GO 91826363 IC50 = 630 nM T03634 C8XL0I 91826394 IC50 = 1400 nM T03634 CD0W7N 91971372 IC50 = 210 nM T03634 C9WB3G 95828281 IC50 = 740 nM T03634 CJ4MO9 95991007 IC50 = 18000 nM T03634 CB19IE 102358573 IC50 = 323 nM T03634 C89GTS 113207960 IC50 = 25370 nM T03634 C7ZLK4 113207965 IC50 = 3390 nM T03634 CGUK73 117098446 IC50 = 39550 nM T03634 CPB3K7 118626392 IC50 = 1000 nM T03634 CZ07JN 118626421 IC50 = 64000 nM T03634 CTF52P 118626429 IC50 = 5000 nM T03634 C9OD6I 118626439 IC50 = 15000 nM T03634 CBQI47 118626440 IC50 = 7400 nM T03634 CA3Q1L 118626445 IC50 = 2000 nM T03634 CD1L7R 118626450 IC50 = 3000 nM T03634 C4H3GM 118633152 IC50 = 7500 nM T03634 CT31MB 118633154 IC50 = 3000 nM T03634 CU95AV 118740117 IC50 = 32000 nM T03634 CFMJ96 119081417 IC50 = 130 nM T03634 C8AZ4C 119081691 IC50 > 20000 nM T03634 CUWX94 119081692 IC50 = 560 nM T03634 C4JN5Q 121237855 IC50 = 120 nM T03634 C4AU0X 121237856 IC50 = 10600 nM T03634 C7A2UY 121237857 IC50 = 650 nM T03634 CBN53Q 121271705 IC50 = 4100 nM T03634 CGBI67 121271742 EC50 = 1900 nM T03634 CPU76D 121271756 IC50 = 250 nM T03634 CN4X9G 121271781 IC50 = 33 nM T03634 CB83MK 121271792 EC50 = 300 nM T03634 C0F6MH 121277645 IC50 = 120000 nM T03634 C0FA3C 121277864 EC50 = 3400 nM T03634 CP1NH2 121277975 IC50 = 3.4 nM T03634 C0XVY8 121277987 EC50 = 1200 nM T03634 CHO97R 121277993 IC50 = 130 nM T03634 COW87E 121278062 IC50 = 110 nM T03634 C1PGY8 121278155 IC50 = 240 nM T03634 C3GD2W 121335190 IC50 > 20000 nM T03634 CECP26 121335281 IC50 > 20000 nM T03634 C8YE5F 121365519 IC50 = 1.5 nM T03634 C4UHQ1 121372691 IC50 = 150 nM T03634 C46MHD 121372830 IC50 = 2 nM T03634 C34YHN 121372887 IC50 = 410 nM T03634 CL67ME 121372914 IC50 = 120 nM T03634 CQ8ZL9 121372939 IC50 = 320 nM T03634 C3I8SV 121372947 IC50 = 1 nM T03634 CVO7B2 121373072 IC50 = 4.7 nM T03634 C57GXL 121373316 IC50 = 1 nM T03634 C04UKS 121373365 IC50 = 1.2 nM T03634 CDH8M4 121373418 IC50 = 1.1 nM T03634 C1TK3U 121373476 IC50 = 1800 nM T03634 C2V6AX 121373769 IC50 = 3.1 nM T03634 C47QXT 121376807 IC50 = 20 nM T03634 C9XWC0 121376818 IC50 = 31 nM T03634 C0QKG5 121376850 IC50 = 4.3 nM T03634 CP6R5B 121382912 IC50 = 46 nM T03634 CVY6B3 122191330 IC50 = 5370 nM T03634 C1EGJ9 122664496 IC50 = 51000 nM T03634 CWJD15 122705990 IC50 = 1710 nM T03634 C5Z9EY 127025709 IC50 > 100000 nM T03634 CNX2L1 127026318 IC50 > 100000 nM T03634 CDA04U 127026319 IC50 > 100000 nM T03634 CP52CH 127027538 IC50 > 10000 nM T03634 C0E7IG 127029904 IC50 > 10000 nM T03634 CT19QO 127029905 IC50 = 1500 nM T03634 C3IJM2 127032947 IC50 = 500000 nM T03634 CT5H3K 127034116 IC50 = 5000 nM T03634 CS56IU 127035170 IC50 = 500000 nM T03634 C6BT3U 127048317 IC50 = 620 nM T03634 C9DY4Z 127048318 IC50 = 670 nM T03634 CEN16G 127049286 IC50 = 900 nM T03634 C9C0MB 127049631 IC50 = 1900 nM T03634 C8MXQ7 127049932 IC50 = 6500 nM T03634 C12KXI 127051477 IC50 = 3400 nM T03634 C5EYK2 127053005 IC50 = 530 nM T03634 CG6AY7 127053006 IC50 = 5000 nM T03634 CY6ZE0 131955089 IC50 = 15 nM T03634 CN62BM 131955090 IC50 = 59 nM T03634 CGNQ49 132168874 IC50 = 170 nM T03634 CHC6A0 132168907 IC50 = 58 nM T03634 CRV1I6 132168917 IC50 = 2.4 nM T03634 CB4X0G 132169005 IC50 = 69 nM T03634 CX9U1Y 132169030 IC50 = 120 nM T03634 CO7QW0 132169133 IC50 = 24 nM T03634 CD8SE7 132169397 IC50 = 69 nM T03634 CG4X6Z 132169416 IC50 = 42 nM T03634 CV8F3O 132169466 IC50 = 90 nM T03634 C7EHB4 132169581 IC50 = 13 nM T03634 CI3HC8 132169624 IC50 = 9.5 nM T03634 CF7H3C 132169928 IC50 = 450 nM T03634 C6HQ0I 132181409 IC50 = 34 nM T03634 C2S4IT 132181414 IC50 = 3.6 nM T03634 C3MV7Y 132181499 IC50 = 5 nM T03634 CM2K6Z 132181651 IC50 = 69 nM T03634 CZW36J 132181706 IC50 = 47 nM T03634 CVZ87Y 132181707 IC50 = 20 nM T03634 CXVW94 132181717 IC50 = 38 nM T03634 CG13LT 132186451 IC50 = 38 nM T03634 CGC84J 132186467 IC50 = 65 nM T03634 CB23YA 132186468 IC50 = 31 nM T03634 C06KYU 132186469 IC50 = 1.2 nM T03634 CI56DE 132186470 IC50 = 81 nM T03634 COK17B 132186514 IC50 = 130 nM T03634 CE3H2T 132186523 IC50 = 1.2 nM T03634 CG5SN9 132186583 IC50 = 120 nM T03634 CN90OX 132186586 IC50 = 30 nM T03634 CAR2X5 132186700 IC50 = 3.3 nM T03634 C5A3QS 132186701 IC50 = 2.8 nM T03634 CKY07I 132186706 IC50 = 79 nM T03634 C4DOU1 132186760 IC50 = 90 nM T03634 CFB2X6 132186767 IC50 = 23 nM T03634 CM6K0J 132186772 IC50 = 13 nM T03634 CL29US 132186773 IC50 = 27 nM T03634 CC6PW8 132186817 IC50 = 31 nM T03634 CUH7W8 132186890 IC50 = 3.3 nM T03634 C31EOG 132275014 IC50 = 19 nM T03634 CGDN94 132275066 IC50 = 0.94 nM T03634 CL1FY9 132451787 IC50 = 1.4 nM T03634 COR87Y 134812725 IC50 = 140 nM T03634 CBF35S 134812726 IC50 = 2200 nM T03634 C3J8KX 134812727 IC50 = 146 nM T03634 C8IDE3 134812728 IC50 = 40 nM T03634 CS7WX6 134821995 IC50 > 20000 nM T03634 CI2AM1 134828588 IC50 = 2450 nM T03634 CV4X7R 135566898 Ki = 7150 nM T03634 CU2F1G 135566900 Ki = 5120 nM T03634 CW94QO 136226511 Ki = 5590 nM T03634 C60DNA 137250528 IC50 = 43 nM T03634 CO71RI 137285009 IC50 > 10000 nM T03634 CS9MR6 137285011 IC50 > 10000 nM T03634 CI1WA0 137319664 IC50 = 130 nM T03634 C53KAO 137631500 IC50 = 300 nM T03634 CA2VS4 137631629 IC50 = 500 nM T03634 C0Y3UF 137631784 IC50 = 740 nM T03634 CUE7F1 137631875 IC50 = 76 nM T03634 C25OZB 137632559 IC50 = 1400 nM T03634 C9XVL1 137635109 IC50 = 260 nM T03634 CM9P2A 137635443 IC50 = 2.2 nM T03634 C0D1LR 137635790 IC50 = 61 nM T03634 CQT3A9 137636309 IC50 > 100000 nM T03634 CYZJ80 137636683 IC50 = 160 nM T03634 C7NZ4E 137637179 IC50 = 330 nM T03634 CT2D8X 137638314 IC50 = 580 nM T03634 CRN21V 137638824 IC50 = 650 nM T03634 CJG6R8 137640750 IC50 = 90 nM T03634 C0SYB2 137640929 IC50 = 170 nM T03634 COK20S 137641504 IC50 = 200 nM T03634 C01BVT 137642411 IC50 = 450 nM T03634 COY3A6 137642659 IC50 = 920 nM T03634 C0R3FG 137646519 IC50 = 39 nM T03634 CWJ7N5 137647079 IC50 = 690 nM T03634 CJ9UI7 137647118 IC50 = 31 nM T03634 CXD50J 137647775 IC50 = 2500 nM T03634 C89VWP 137649346 IC50 = 310 nM T03634 C85QNS 137649815 IC50 = 470 nM T03634 CKN60B 137649822 IC50 = 500 nM T03634 CO7K6Y 137649906 IC50 = 360 nM T03634 C4Y8HV 137650663 IC50 = 310 nM T03634 CE42GP 137650954 IC50 = 400 nM T03634 CSV15U 137650957 IC50 = 540 nM T03634 CV9F6J 137651164 IC50 = 1500 nM T03634 CHN7A8 137652035 IC50 = 200 nM T03634 CCZD32 137652808 IC50 = 140 nM T03634 CHU2W4 137653154 IC50 > 30000 nM T03634 C7Y6IH 137653562 IC50 = 210 nM T03634 CL1V9T 137654008 IC50 = 240 nM T03634 C3OX9R 137655043 IC50 = 2400 nM T03634 CM7Y4D 137655923 IC50 = 980 nM T03634 C5B7LO 137656022 IC50 = 780 nM T03634 CX35DY 137656164 IC50 = 240 nM T03634 C8BP5R 137656667 IC50 = 310 nM T03634 CW9C8L 137657087 IC50 = 400 nM T03634 C5TEY3 137657620 IC50 = 1300 nM T03634 CE3CQ5 137659158 IC50 = 130 nM T03634 CQ6XB7 139030526 IC50 > 100000 nM T03634 CYQ79A 139382567 IC50 = 81 nM T03634 C9IDO1 141736322 IC50 = 1860 nM T03634 CWM80Y 141736350 IC50 = 33850 nM T03634 C7YR4W 141736357 IC50 = 690 nM T03634 C8ZQ2U 141736359 IC50 = 140 nM T03634 CV7G1U 141736363 IC50 = 19840 nM T03634 C5VNM4 141736367 IC50 = 37 nM T03634 C1P3TL 141736369 IC50 = 2070 nM T03634 C5O6SU 141736374 IC50 = 1000 nM T03634 C4SCT9 141736375 IC50 = 2800 nM T03634 CB68VY 141736376 IC50 = 3520 nM T03634 C4NHG5 141736379 IC50 = 4050 nM T03634 C1V4ND 141736380 IC50 = 1440 nM T03634 CM6ZO2 141736388 IC50 = 32640 nM T03634 C7SQ8T 141736403 IC50 = 6360 nM T03634 C0TB5Z 141736419 IC50 = 26190 nM T03634 C0RV7I 141736434 IC50 = 170 nM T03634 C5UAO0 145949218 IC50 = 2330 nM T03634 COT05Q 145949275 IC50 = 1670 nM T03634 C4IXO6 145950180 IC50 = 290 nM T03634 CIA1W6 145950654 IC50 = 1890 nM T03634 C96NCH 145950955 IC50 = 770 nM T03634 C03SNP 145951746 IC50 = 3890 nM T03634 CYS60Q 145951844 IC50 = 2990 nM T03634 C3ZV1O 145952497 IC50 = 1690 nM T03634 C6LO5F 145953516 IC50 = 2740 nM T03634 C2YR6U 145953602 IC50 = 1690 nM T03634 CSR9N7 145953663 IC50 = 2560 nM T03634 CTE74G 145954441 IC50 = 1000 nM T03634 CR6OX1 145954766 IC50 = 2650 nM T03634 C2Y3ZT 145955733 IC50 = 2330 nM T03634 CNQD23 145956474 IC50 = 4700 nM T03634 CCNU52 145956492 IC50 = 2470 nM T03634 C1NSW8 145956646 IC50 > 50000 nM T03634 C4AI2J 145957252 IC50 = 6560 nM T03634 CN5YO3 145957310 IC50 = 160 nM T03634 CN7G8J 145957486 IC50 = 2480 nM T03634 C7C5WL 145958595 IC50 = 650 nM T03634 C2TH1N 145959035 IC50 = 4840 nM T03634 CE5FW8 145959058 IC50 = 8500 nM T03634 CW6O3D 145959144 IC50 > 50000 nM T03634 CCP03T 145959259 IC50 = 2810 nM T03634 CDNG83 145959505 IC50 = 2060 nM T03634 C4Y0PN 145967100 IC50 = 280 nM T03634 C3BSE8 145971523 IC50 = 1560 nM T03634 C5CXR4 145971749 IC50 = 1960 nM T03634 CIU53N 145972433 IC50 = 7090 nM T03634 CEY8P5 145972450 IC50 = 3390 nM T03634 CNU4O9 145972623 IC50 = 0.9 nM T03634 CC8LU2 145972824 IC50 = 240 nM T03634 CD4A3Y 145973334 IC50 = 650 nM T03634 CR3E9H 145973362 IC50 = 21580 nM T03634 C37UVN 145973834 IC50 = 4110 nM T03634 CP49HN 145974181 IC50 = 180 nM T03634 CA85TK 145975493 IC50 = 190 nM T03634 CZV20H 145976144 IC50 = 7700 nM T03634 CQN6G3 155532286 IC50 > 20000 nM T03634 C0QV9U 155534567 IC50 > 20000 nM T03634 C95OQP 155536635 IC50 = 1200 nM T03634 C62EMT 155540785 IC50 > 20000 nM T03634 C7VRN8 155541456 IC50 > 20000 nM T03634 C5NU8A 155564453 IC50 > 20000 nM T03634 D00DXI 135566302 IC50 = 5000 nM T03634 D03XXT 72201027 IC50 = 30 nM T03634 D09HBR 135566899 Ki = 2180 nM T03634 D0H3TC 54669868 IC50 = 28100 nM T03634 D0J3JI 90488984 IC50 = 440 nM T03634 D0O2RX 71624782 IC50 = 2480 nM T03634 D0YL8Z 1285940 IC50 = 2.6 nM T66237 D03KZM 216237 Ki = 0.43 nM T66237 D08FJL 16681432 EC50 = 170 nM T66237 D09GOS 2812 IC50 = 15848.93 nM T66237 D0D8XY 5311010 Ki = 330 nM T66237 D0F4NS 119369 Ki = 9.42 nM T66237 D0K8KX 5280343 IC50 = 15200 nM T66237 D0M3FJ 439302 EC50 = 7.3 nM T66237 D0N4OW 644077 EC50 = 0.05 nM T66237 D0U7SH 5311065 EC50 = 0.2 nM T66237 D0VU2X 151171 Ki = 0.36 nM T66237 D04QZI 11340891 Ki = 950 nM T66237 D06VWL 10298385 EC50 = 24 nM T66237 D07EEN 172997 IC50 = 1 nM T66237 D09WYL 11634973 Ki = 3981.07 nM T66237 D0L6XQ 11157078 IC50 = 34 nM T66237 D0LI1C 44469321 IC50 > 30000 nM T66237 D0S3YN 53330936 EC50 = 2630.27 nM T66237 D0SY9B 9895468 Ki = 290 nM T66237 D02RDE 9939929 IC50 = 20 nM T66237 D03RYS 5311500 EC50 = 0.7 nM T66237 D08ORO 114904 Ki > 10000 nM T66237 D08PAC 6918320 Ki = 37000 nM T66237 D0A1KU 11683187 IC50 = 1530 nM T66237 D0AV0O 3038506 Ki = 91.9 nM T66237 D0I8ZZ 60943 Ki = 178 nM T66237 D0Q8RX 9872389 Ki = 590 nM T66237 CY4WG9 3793 IC50 = 6000 nM T66237 C0R7SI 449224 EC50 = 3.5 nM T66237 C5F1ST 1103817 Ki = 2500 nM T66237 C7AD6Y 5034737 Ki = 2460 nM T66237 CQB93O 5306925 Ki = 507 nM T66237 COSN76 6918573 EC50 = 58 nM T66237 C93WRU 9690136 Ki > 10000 nM T66237 C5E3XU 9799174 IC50 = 390 nM T66237 C4PY7Z 9801970 IC50 = 390 nM T66237 CC07MW 9807249 Ki = 0.9 nM T66237 CC24MQ 9807250 Ki = 15 nM T66237 CO3SD6 9811830 EC50 = 154.88 nM T66237 CML46C 9824954 EC50 = 1.67 nM T66237 C57WZH 9826033 IC50 = 20 nM T66237 CS8Q6R 9826254 IC50 = 3.2 nM T66237 CW8ZA7 9828129 IC50 = 8 nM T66237 C6OV5R 9829108 IC50 > 1000 nM T66237 CK4UY8 9848300 IC50 = 8 nM T66237 CQYU70 9849525 Ki = 5 nM T66237 CZ3M1F 9850567 IC50 = 13 nM T66237 C0K2IJ 9851013 IC50 = 5.2 nM T66237 CU1W4L 9868852 IC50 = 296 nM T66237 C17GIC 9869993 IC50 = 11 nM T66237 CA7RO2 9871426 IC50 = 7 nM T66237 CGTK84 9874047 IC50 = 2.6 nM T66237 C6D0OX 9887157 IC50 = 933 nM T66237 CA2J5M 9888109 IC50 = 91.5 nM T66237 C8LR0K 9889904 IC50 = 413 nM T66237 CT4S6Q 9910527 IC50 = 475 nM T66237 CDFI62 9915472 IC50 = 4 nM T66237 CRM93H 9931699 IC50 = 183 nM T66237 CPBC63 9935694 IC50 = 210 nM T66237 C9DAQ2 9935969 IC50 = 44 nM T66237 C1C6HA 9937535 IC50 = 341 nM T66237 COUA25 9938406 Ki = 130 nM T66237 C4V2XT 9939024 IC50 = 2 nM T66237 CH2K5E 9954641 EC50 = 47 nM T66237 CNJ81W 9959174 EC50 = 1.8 nM T66237 CD4B6A 9959838 IC50 = 7.5 nM T66237 CW9U3E 9961036 IC50 = 11.5 nM T66237 CK97LP 9974701 IC50 = 18 nM T66237 CIE8X5 9981665 Ki = 5600 nM T66237 C9J4MZ 10003306 IC50 = 1.5 nM T66237 CFO98G 10043741 IC50 = 9 nM T66237 CBI6W4 10098338 IC50 = 1.7 nM T66237 CT7SZ8 10119966 Ki = 21 nM T66237 C1C4SX 10142915 Ki = 2470 nM T66237 C98HVI 10144208 Ki = 8520 nM T66237 C68ZRW 10156521 IC50 = 2000 nM T66237 CRQW02 10162731 EC50 = 2.3 nM T66237 CL71MC 10164478 Ki = 1780 nM T66237 C2NEU9 10165683 Ki = 8890 nM T66237 C7VW8K 10187283 Ki = 585 nM T66237 CZPR64 10187625 EC50 = 890 nM T66237 C91QFB 10206789 EC50 = 4.7 nM T66237 CV7A0N 10206901 Ki = 6930 nM T66237 CPE3F8 10208389 Ki = 14400 nM T66237 CP7N1H 10231366 IC50 = 4 nM T66237 CV2Z3J 10278394 Ki = 4850 nM T66237 CH2XI7 10279928 IC50 = 6 nM T66237 C8UK7I 10281429 EC50 = 10 nM T66237 C72BJX 10282736 EC50 = 1100 nM T66237 C4LU8J 10303620 Ki = 979 nM T66237 C52SOK 10304617 Ki = 1920 nM T66237 CF6A5Y 10322392 IC50 = 67 nM T66237 CW50TU 10345610 EC50 = 215 nM T66237 CPA89S 10390899 IC50 = 6.8 nM T66237 C06SVZ 10392505 IC50 = 7 nM T66237 CTWG68 10411308 Ki = 0.57 nM T66237 CKD75B 10414302 Ki = 3.2 nM T66237 C1OIW6 10416272 Ki > 3000 nM T66237 C8DWH6 10456892 EC50 = 13 nM T66237 C5JSO3 10459252 IC50 = 2.7 nM T66237 C1Z3WY 10461417 IC50 = 11 nM T66237 CR6VX2 10483105 Ki = 181 nM T66237 C9H8WU 10495509 IC50 = 4.1 nM T66237 C8WK5N 10498917 IC50 = 13 nM T66237 CY58RQ 10503858 IC50 = 2.1 nM T66237 C6WXS4 10519373 IC50 = 35 nM T66237 C6PS5H 10569977 IC50 = 8.8 nM T66237 C79NZO 10570880 IC50 = 13 nM T66237 CM7Q1K 10578000 IC50 = 80 nM T66237 CFP17Y 10578460 IC50 = 60 nM T66237 C2Z7RB 10587836 IC50 = 180 nM T66237 CS39QY 10591515 IC50 = 320 nM T66237 CQEP07 10595255 IC50 = 120 nM T66237 CR01ZV 10603742 IC50 > 10000 nM T66237 CSP1C3 10626339 IC50 = 80 nM T66237 CD9ZU1 10642447 IC50 = 5 nM T66237 C5NIU8 10648029 IC50 = 0.5 nM T66237 CLXT94 10672170 IC50 = 1.9 nM T66237 C8VB3L 10673295 IC50 = 2 nM T66237 CZKU73 10673699 IC50 = 8.3 nM T66237 C4RAN8 10691737 IC50 = 16 nM T66237 CYE0I7 10696913 IC50 = 1.9 nM T66237 CRAC01 10710850 IC50 = 1000 nM T66237 C96EYF 10711405 IC50 = 18 nM T66237 CCU35N 10715974 Ki = 7.56 nM T66237 CH84ZE 10719289 IC50 = 4 nM T66237 CEC70P 10737018 IC50 = 22 nM T66237 C6FW1B 10737785 IC50 = 51 nM T66237 CR8QV4 10742418 IC50 = 1 nM T66237 CL1N4A 10743786 IC50 = 0.7 nM T66237 CODM17 10758700 IC50 = 34 nM T66237 CU4EL3 10766720 IC50 = 2 nM T66237 CCHY18 10784361 IC50 = 210 nM T66237 C4GTY9 10814200 IC50 = 4.2 nM T66237 C5GB4F 10831068 IC50 = 5.9 nM T66237 CA9C1V 10831734 IC50 = 7.5 nM T66237 C2TL5U 10837633 IC50 = 4 nM T66237 C58XOT 10840974 IC50 = 50 nM T66237 C3U6QA 10863737 Ki = 11100 nM T66237 CQJ52W 10873853 Ki = 8170 nM T66237 C1WD7P 10907482 Ki = 6650 nM T66237 CI8AQ1 10929819 Ki = 14300 nM T66237 CMZ2W9 10984131 IC50 = 14 nM T66237 CBOS05 11016093 Ki = 4430 nM T66237 C9GX3E 11070458 IC50 = 980 nM T66237 CFL2P5 11092056 Ki = 10200 nM T66237 CDF9W0 11144861 Ki = 7370 nM T66237 C4C8QJ 11158261 IC50 = 9 nM T66237 CZWJ61 11167861 IC50 = 30 nM T66237 C4JKH8 11190868 IC50 = 30 nM T66237 C0FJM7 11194023 Ki = 568 nM T66237 C6D3UR 11237434 EC50 = 265 nM T66237 C2PE4M 11238362 IC50 = 71 nM T66237 CB43VY 11239468 IC50 = 30 nM T66237 CO3A5Z 11240155 Ki = 36.8 nM T66237 CC0KT1 11251777 Ki = 621 nM T66237 CUED54 11257380 Ki > 10000 nM T66237 CU1E4A 11261339 IC50 = 120 nM T66237 C9Q7RV 11262100 IC50 = 80 nM T66237 CE0DX4 11269308 IC50 > 10000 nM T66237 CZ0JW9 11270497 IC50 > 10000 nM T66237 C89CZT 11272841 IC50 = 200 nM T66237 C5OTG4 11274745 Ki = 1090 nM T66237 C9T8BV 11286254 Ki = 80 nM T66237 CB6TF8 11297732 Ki = 1067 nM T66237 CTP85J 11317662 IC50 < 10 nM T66237 CFU2E1 11351397 IC50 = 60 nM T66237 CN2YM9 11365307 IC50 = 50 nM T66237 CYJ23D 11384094 Ki = 103 nM T66237 CON43W 11386922 IC50 = 20 nM T66237 CPND10 11389106 Ki = 24.7 nM T66237 CHRT50 11397211 IC50 < 10 nM T66237 CEM1X7 11400547 Ki = 1386 nM T66237 C93VQG 11418441 IC50 > 10000 nM T66237 CPG63Z 11422294 IC50 = 8 nM T66237 CG0Q5O 11432362 IC50 = 53 nM T66237 CR4N5I 11465834 Ki = 39.81 nM T66237 CM83DS 11468862 Ki = 11170 nM T66237 C37TNB 11475469 Ki > 10000 nM T66237 CN14VO 11476070 IC50 > 10000 nM T66237 C9SY7Q 11486351 Ki = 6400 nM T66237 COC7Q9 11488952 Ki = 5011.87 nM T66237 CIS2N6 11490514 IC50 = 1 nM T66237 CZ3PM4 11490613 IC50 = 6 nM T66237 CR5SH4 11502419 Ki > 10000 nM T66237 C5PU0J 11538526 Ki > 10000 nM T66237 CQ96XZ 11569194 Ki = 1258.93 nM T66237 C60DKW 11569672 Ki > 79432.82 nM T66237 CM15EB 11574636 Ki > 10000 nM T66237 CG7CL9 11578939 EC50 = 281.84 nM T66237 CU9F1K 11618185 Ki > 10000 nM T66237 CFPR21 11625088 Ki > 10000 nM T66237 CQ4SX5 11667812 Ki > 10000 nM T66237 CY0HE4 11677610 IC50 > 100000 nM T66237 CIC93G 11740743 Ki = 2.68 nM T66237 CVWH18 11757222 IC50 = 15 nM T66237 COJ27D 11763684 IC50 = 10 nM T66237 CJ7BP8 11792631 IC50 = 19 nM T66237 C6XGN2 11793558 IC50 = 31 nM T66237 C91CIO 11815584 Ki = 50 nM T66237 C8GC2P 11854507 IC50 > 100000 nM T66237 CEX2I5 14182908 Ki = 400000 nM T66237 C4CTD2 14257660 EC50 = 0.4467 nM T66237 C1E4BW 15298022 IC50 = 510 nM T66237 CEI74X 15307998 IC50 = 9 nM T66237 CIDT94 15307999 IC50 = 19 nM T66237 CMP0I2 15308000 IC50 = 0.7 nM T66237 C06DHE 15416417 Ki = 4.87 nM T66237 CU3M1I 15416418 Ki = 8.3 nM T66237 C9HNQ6 15896091 EC50 = 140 nM T66237 C0WNE9 15896092 EC50 = 180 nM T66237 CA3B4L 15896094 EC50 = 37 nM T66237 CTEW91 15951937 Ki > 27000 nM T66237 C1SKJ3 15953022 Ki = 9308 nM T66237 CHU5E4 16051933 Ki = 5 nM T66237 C3TX0W 18759802 EC50 = 210 nM T66237 CUX27F 18759808 EC50 = 150 nM T66237 C2U0JN 18759812 EC50 = 140 nM T66237 C0OT2Q 18759822 EC50 = 120 nM T66237 CFOU06 18759824 EC50 = 100 nM T66237 C8CY9A 19607875 Ki = 870 nM T66237 CGDY68 19608069 Ki = 21 nM T66237 CJ8MC9 19699060 IC50 = 140 nM T66237 CGC20J 19699093 IC50 = 130 nM T66237 C65CTX 19699097 IC50 = 71 nM T66237 CY89CI 19699133 IC50 = 150 nM T66237 C6TKQ8 20825285 IC50 = 30 nM T66237 C84GPV 21083206 EC50 = 140 nM T66237 CX5H6M 21083210 EC50 = 180 nM T66237 C8R5PD 21083212 EC50 = 82 nM T66237 C7D8XH 21467167 IC50 = 5 nM T66237 C59LDI 22405322 IC50 = 58 nM T66237 CUD2I8 22405325 IC50 = 15000 nM T66237 CGD49J 22405327 IC50 = 96 nM T66237 CW7O1M 22405331 IC50 = 2500 nM T66237 C10PQM 23505561 IC50 = 170 nM T66237 CE4Z6R 23598556 IC50 = 550 nM T66237 CEOZ91 23598560 IC50 = 29 nM T66237 C71XOU 23598595 IC50 = 14 nM T66237 CBRI52 23598597 IC50 = 110 nM T66237 CJ8Z6N 23598598 IC50 = 8 nM T66237 CM1F7K 23598600 IC50 = 39 nM T66237 CP8GK0 23598619 IC50 > 10000 nM T66237 CPZE93 23598641 IC50 = 18 nM T66237 CP64WA 23598642 IC50 = 44 nM T66237 CG20SB 25132666 IC50 = 40 nM T66237 C7C1TG 25132999 IC50 = 1050 nM T66237 CWSF74 25133000 IC50 = 11 nM T66237 C3Q0AD 25133001 IC50 = 730 nM T66237 CM2CP4 25178587 EC50 = 110 nM T66237 C5PHN1 25178591 EC50 = 130 nM T66237 C3WBD7 25178592 EC50 = 820 nM T66237 CS81BP 25178784 EC50 = 270 nM T66237 C65RXN 25178785 EC50 = 100 nM T66237 CG96CK 25178786 EC50 = 390 nM T66237 C8BE6A 25178787 EC50 = 380 nM T66237 C0FH5N 25178959 EC50 = 46 nM T66237 CHA97X 25178960 EC50 = 27 nM T66237 C1E2JZ 25178961 EC50 = 230 nM T66237 C5MV7R 25178962 EC50 = 1700 nM T66237 CWD3Q1 25178963 EC50 = 120 nM T66237 CLD0E7 25180311 EC50 = 30 nM T66237 C1ACZ3 25180507 EC50 = 730 nM T66237 C27WJL 25180508 EC50 = 680 nM T66237 CHV48R 25180509 EC50 = 950 nM T66237 CA9B6P 25180695 EC50 = 350 nM T66237 C5EGS7 25180696 EC50 = 3.2 nM T66237 COJ3F2 25180697 EC50 = 4.3 nM T66237 C5HPT0 25180884 EC50 = 220 nM T66237 CU1OE3 25180885 EC50 = 1000 nM T66237 CM9D7O 25180886 EC50 = 84 nM T66237 CVF12W 25180887 EC50 = 140 nM T66237 C4FLY0 25181104 EC50 = 40 nM T66237 CM1QA7 25181105 EC50 = 10 nM T66237 COC73W 25212177 Ki = 12589.25 nM T66237 CCX14Y 26434734 Ki = 468 nM T66237 CY67HA 42611262 Ki = 251.19 nM T66237 CS04KE 42629368 EC50 = 4.2 nM T66237 CYGN52 42629369 EC50 = 6.3 nM T66237 CMS6P8 44214518 IC50 = 4 nM T66237 CB82ZC 44232512 EC50 = 160 nM T66237 CBV47F 44243143 Ki = 500 nM T66237 CDI2Q4 44247566 IC50 > 31622.78 nM T66237 CVI6Q3 44275104 Ki = 137 nM T66237 CW7JM3 44275447 Ki = 282 nM T66237 CDQ3A6 44294573 Ki = 3.3 nM T66237 C2J8GK 44316235 Ki = 13.7 nM T66237 CIE6Y1 44316236 Ki = 554 nM T66237 C24NQS 44316241 Ki = 245 nM T66237 CS2ZN9 44321415 Ki = 10200 nM T66237 CK2JA7 44325332 Ki = 3.7 nM T66237 CHW9O4 44325345 Ki = 2.8 nM T66237 CS4UM7 44325362 Ki = 1.9 nM T66237 C4STM0 44325363 Ki = 4.2 nM T66237 CXU9H7 44325377 Ki = 17 nM T66237 C1H6JQ 44325505 Ki = 11 nM T66237 CAUJ69 44325531 Ki = 9 nM T66237 CAG0C8 44325538 Ki = 4.2 nM T66237 CK5TS8 44325543 Ki = 10 nM T66237 CE8F7A 44325545 Ki = 18 nM T66237 CH1P8N 44325558 Ki = 5 nM T66237 CP4FH8 44325579 Ki = 3.2 nM T66237 C6OV2D 44325607 Ki = 2.8 nM T66237 CZ0BD9 44325689 Ki = 11 nM T66237 C91EAF 44325691 Ki = 3.7 nM T66237 CO3ZL8 44325695 Ki = 2 nM T66237 CQ6MC5 44325703 Ki = 1.4 nM T66237 C1BA7W 44325704 Ki = 13 nM T66237 CO9Y1C 44325731 Ki = 10 nM T66237 CW23ZH 44325732 Ki = 10 nM T66237 CR4TV5 44325733 Ki = 15 nM T66237 C19AEH 44325766 Ki = 3.7 nM T66237 CD86NE 44325804 Ki = 8 nM T66237 CG8P5Z 44325895 Ki = 25 nM T66237 CM94YJ 44325896 Ki = 40 nM T66237 CV54FN 44325905 Ki = 37 nM T66237 C08ETV 44325915 Ki = 60 nM T66237 C95HKU 44332168 IC50 = 390 nM T66237 CSF89I 44332181 IC50 > 1000 nM T66237 C6NW1Z 44332207 IC50 = 274 nM T66237 CF3QT6 44332208 IC50 = 159 nM T66237 CPF97V 44332209 IC50 = 180 nM T66237 CRL53G 44332212 IC50 > 1000 nM T66237 C5N1TG 44332226 IC50 > 1000 nM T66237 C4UD2C 44332237 IC50 > 1000 nM T66237 CB2VP5 44332238 IC50 > 1000 nM T66237 C98OKM 44332239 IC50 = 0.2 nM T66237 CLJN56 44332261 IC50 > 1000 nM T66237 CA1OL4 44332269 IC50 > 1000 nM T66237 C8L7KE 44332272 IC50 = 380 nM T66237 C0S9TC 44332273 IC50 = 70 nM T66237 CGT2A0 44335241 IC50 = 72 nM T66237 C6HO3T 44335329 IC50 = 5 nM T66237 CO0EQ9 44335343 IC50 = 13 nM T66237 CZ75ET 44335345 IC50 = 10 nM T66237 C23MCR 44335356 IC50 = 28 nM T66237 CONI47 44335357 IC50 = 19 nM T66237 C8VWX6 44335386 IC50 = 26 nM T66237 C92YST 44336379 IC50 = 23 nM T66237 C7X3QZ 44336402 IC50 > 1000 nM T66237 CDTJ17 44336403 IC50 > 1000 nM T66237 CENA29 44336404 IC50 = 20 nM T66237 CM61WN 44336418 IC50 = 10 nM T66237 C7ML9D 44336636 IC50 = 11 nM T66237 CZYV25 44336768 IC50 = 18 nM T66237 CD62CM 44336784 IC50 = 16 nM T66237 C7AU5H 44336791 IC50 > 1000 nM T66237 C2IJS5 44336799 IC50 > 1000 nM T66237 C1TEP7 44351278 Ki = 6.6 nM T66237 CL2R8E 44351441 Ki = 3.7 nM T66237 COE18X 44351500 Ki = 1.5 nM T66237 CJR5B7 44352302 IC50 = 430 nM T66237 CZ60LX 44352757 IC50 = 7 nM T66237 CM4ZJ0 44352767 IC50 = 100 nM T66237 C9UBG4 44352768 IC50 = 16 nM T66237 C2X8GD 44352776 IC50 = 20 nM T66237 CTNY07 44352777 IC50 = 12 nM T66237 CT3Z9C 44352783 IC50 = 8 nM T66237 CVK34U 44352796 IC50 = 85 nM T66237 CLA4U8 44352804 IC50 = 15 nM T66237 CH41KQ 44357890 IC50 = 0.95 nM T66237 COUJ27 44374802 IC50 = 3.4 nM T66237 CVR8H4 44374839 IC50 = 220 nM T66237 CY4TC0 44375638 Ki = 1 nM T66237 CMI9C7 44377521 IC50 = 550 nM T66237 CQ50CE 44377836 IC50 = 50 nM T66237 CVU70Y 44377837 IC50 = 190 nM T66237 C9WO6P 44377894 IC50 = 180 nM T66237 CXG0R3 44377903 IC50 = 15 nM T66237 C5HWR0 44377961 IC50 = 12 nM T66237 CV1BR7 44378675 IC50 = 8.8 nM T66237 CU6CL9 44378702 IC50 = 2 nM T66237 CPWO06 44378703 IC50 = 2.1 nM T66237 C6TX2Q 44378719 IC50 = 1.3 nM T66237 C6OTD5 44378885 IC50 = 7 nM T66237 C1NA5W 44378886 IC50 = 14.8 nM T66237 CYBX91 44382370 Ki = 1.1 nM T66237 CH47GO 44382498 Ki = 0.99 nM T66237 CKL2S9 44382499 Ki = 1 nM T66237 CJBV97 44386548 IC50 < 10 nM T66237 C9E5JO 44393911 EC50 = 200 nM T66237 CDK52W 44393912 EC50 = 100 nM T66237 CZ4UB9 44393941 EC50 = 570 nM T66237 C9JBI3 44393965 EC50 = 1300 nM T66237 CGW9Z6 44393998 EC50 = 1800 nM T66237 CUS19Z 44394044 EC50 = 230 nM T66237 C05DOG 44394045 EC50 = 1200 nM T66237 CZ4B0C 44394063 EC50 = 1800 nM T66237 C9BH3V 44404614 IC50 = 300 nM T66237 CF80BP 44433360 IC50 = 1214 nM T66237 CS8M2O 44433363 IC50 = 11 nM T66237 CLBA10 44433367 IC50 = 34 nM T66237 CCI04H 44433372 IC50 = 1000 nM T66237 C9BDH6 44433375 IC50 = 1000 nM T66237 CF2U3N 44444760 IC50 = 76 nM T66237 CR8OX5 44444761 IC50 > 10000 nM T66237 C1YR6A 44444762 IC50 = 36 nM T66237 CLE7W0 44466239 IC50 > 31622.78 nM T66237 CKA3S0 44467347 IC50 > 31622.78 nM T66237 C2N8FY 44520848 EC50 = 2.4 nM T66237 C91HXT 44520849 EC50 = 0.99 nM T66237 C3HP9Y 44520850 EC50 = 1 nM T66237 CZ5E2V 44520851 EC50 = 0.98 nM T66237 CMGE92 44520852 EC50 = 1 nM T66237 CVA7R2 44520853 Ki = 20 nM T66237 C1U0RY 44520854 Ki = 19 nM T66237 CHE1Y6 44520855 Ki = 5.6 nM T66237 CCW48G 44520856 Ki = 16 nM T66237 CK7O1L 44520857 Ki = 10 nM T66237 C6TOE7 44520858 Ki = 11 nM T66237 CQF23X 44520859 Ki = 7.4 nM T66237 CFD98V 44520860 Ki = 14 nM T66237 CJCB39 44520861 Ki = 3.4 nM T66237 CTVS34 44520862 Ki = 11 nM T66237 CT5A0C 44520863 Ki = 11 nM T66237 CPR8F2 44520864 Ki = 11 nM T66237 CR7Y8G 44520865 Ki = 12 nM T66237 CUN6S2 44520866 Ki = 27 nM T66237 CY61JM 44520867 Ki = 33 nM T66237 CW9RI7 44520868 Ki = 18 nM T66237 CRIF68 44520869 Ki = 53 nM T66237 C1JN3D 44520870 Ki = 22 nM T66237 C8X5FQ 44520871 Ki = 11 nM T66237 C2SDC4 44563370 EC50 = 50 nM T66237 CZF2R4 44563371 EC50 = 20 nM T66237 CPI04M 44563579 EC50 = 2.1 nM T66237 CMG70R 44577936 Ki = 500 nM T66237 CZD7E3 44577937 Ki = 160 nM T66237 C0HXR2 44577938 Ki > 10000 nM T66237 COP3Q0 44577939 Ki > 10000 nM T66237 C10ZLO 44577981 Ki > 10000 nM T66237 CED75W 44577983 Ki > 10000 nM T66237 C1E6GX 44577984 Ki > 10000 nM T66237 C6R0AW 44578010 Ki > 10000 nM T66237 CLCK14 44579399 Ki > 10000 nM T66237 C6OK3X 44579400 Ki > 10000 nM T66237 C0IHE7 44579401 Ki > 10000 nM T66237 CU31MF 44579402 Ki > 10000 nM T66237 CXOJ34 44579441 Ki > 10000 nM T66237 CMW6Q7 44579442 Ki = 1000 nM T66237 CM7HN8 44581240 Ki = 501.19 nM T66237 CG68XT 44581241 Ki = 1258.93 nM T66237 CC5AT2 44581242 Ki = 251.19 nM T66237 C4FZQ9 44581266 Ki = 63.1 nM T66237 CZ9KU4 44589838 EC50 = 1.8 nM T66237 C8R7ZF 44589839 Ki = 9.2 nM T66237 C8YJ1I 44589840 Ki = 21 nM T66237 C6MRI9 44589841 Ki = 18 nM T66237 C58BYM 44589842 Ki = 11 nM T66237 CR32JK 44589843 Ki = 9.1 nM T66237 CF5LG2 44589844 Ki = 6 nM T66237 CD64HU 44589892 Ki = 20 nM T66237 C4OT3X 44589893 EC50 = 3.13 nM T66237 C4CX0I 44589894 EC50 = 1.25 nM T66237 C7DT5U 44589895 Ki = 16 nM T66237 C91MTZ 44589946 Ki = 14 nM T66237 C6J3KX 44589947 Ki = 11 nM T66237 C49UZD 44589948 Ki = 200 nM T66237 CTA89E 44589949 Ki = 170 nM T66237 CSZ70I 45103785 Ki = 3400 nM T66237 CK4XM7 45103786 Ki > 5000 nM T66237 C6LX7B 46225023 Ki > 10000 nM T66237 C48JOB 46225048 Ki > 10000 nM T66237 CX2S6L 46225049 Ki > 10000 nM T66237 C70FCZ 46225050 Ki > 10000 nM T66237 CIM9Y4 46225051 Ki > 10000 nM T66237 CZ36XD 46225079 Ki > 10000 nM T66237 CA6DS1 46225080 Ki > 10000 nM T66237 COT65W 46225081 Ki > 10000 nM T66237 C53ZIX 46225082 Ki > 10000 nM T66237 CFLW87 46225083 Ki > 10000 nM T66237 C7A8DU 46225116 Ki > 10000 nM T66237 C4E8NX 46225117 Ki > 10000 nM T66237 C3W6VI 46225118 Ki = 2770 nM T66237 CT8LO5 46225153 Ki = 1190 nM T66237 C98EDC 46233065 Ki > 1000 nM T66237 C4K7AV 46830094 Ki = 2400 nM T66237 CH4F6K 46830095 Ki = 2300 nM T66237 CNU72P 46830096 Ki = 2830 nM T66237 C0EMW2 46884414 Ki > 10000 nM T66237 C3FUB6 46884437 Ki > 10000 nM T66237 CM0RI1 46884438 Ki > 10000 nM T66237 C4DP6I 46884439 Ki > 10000 nM T66237 CXTE54 46884441 Ki > 10000 nM T66237 C27WFG 46884478 Ki > 10000 nM T66237 C3U2WD 46884479 Ki > 10000 nM T66237 CB8WK2 46884480 Ki = 343000 nM T66237 CIS28Y 46890052 Ki = 63 nM T66237 CWH0O5 46890053 Ki = 2380 nM T66237 CG35DC 46890054 Ki = 2090 nM T66237 CQPV07 46890055 Ki = 2470 nM T66237 CMBS14 46890099 Ki = 1890 nM T66237 CLFP63 46890100 Ki = 770 nM T66237 CRP96J 46890101 Ki = 130 nM T66237 CNJB38 46890102 Ki > 2500 nM T66237 CE84XQ 46890151 Ki > 2500 nM T66237 C8Y6ET 46890152 Ki = 124 nM T66237 C8CXM4 46890153 Ki = 233 nM T66237 CZWV30 46890154 Ki = 171 nM T66237 CY3P8V 46890184 Ki = 36.5 nM T66237 C60CEY 46890185 Ki = 21 nM T66237 CO4CU1 46890186 Ki = 60.6 nM T66237 CJD1S7 46890187 Ki = 133 nM T66237 CLON70 46890214 Ki = 176 nM T66237 CN76SA 46890215 Ki = 39.2 nM T66237 C0AZT4 46890216 Ki > 2550 nM T66237 CJ0AM6 46890217 Ki > 2550 nM T66237 C1DG3H 46890258 Ki > 2550 nM T66237 CJ2L6D 46890259 Ki > 2550 nM T66237 CM70JW 46890260 Ki > 2550 nM T66237 CQWM92 46890261 Ki = 9.2 nM T66237 CC85GR 46890262 Ki = 82 nM T66237 CIC2E8 46890288 Ki = 40 nM T66237 CC75DR 46890289 Ki = 43.4 nM T66237 CW38OV 46890290 Ki = 420 nM T66237 CHFR58 46890438 Ki = 204 nM T66237 CVD95O 46890439 Ki = 3345 nM T66237 COE5S9 46890440 Ki = 54 nM T66237 C0N1MO 46890484 Ki = 1032 nM T66237 CR84PB 46890485 Ki = 478 nM T66237 CA7BO2 46890486 Ki = 1057 nM T66237 CAR94C 46890487 Ki = 82 nM T66237 CEM4L1 46890528 Ki = 107 nM T66237 C2PYH3 46890529 Ki = 1205 nM T66237 CCI0R6 46890530 Ki > 2500 nM T66237 CF83TS 46890531 Ki = 846 nM T66237 C0T5MG 46890569 Ki = 189 nM T66237 C1JSF8 46890570 Ki > 2500 nM T66237 C9QJ5V 46890571 Ki = 713 nM T66237 C83LYU 46890572 Ki = 1170 nM T66237 C1VNK6 46890612 Ki = 30 nM T66237 C2XDO1 46890613 Ki > 2500 nM T66237 CC9E4R 46890614 Ki = 1810 nM T66237 CCM29N 46890615 Ki = 291 nM T66237 C39HAX 46890654 Ki = 556 nM T66237 CQUA46 46890655 Ki > 2500 nM T66237 CLJ2O5 46890656 Ki = 675 nM T66237 CEH20W 46890657 Ki > 2500 nM T66237 CC7Y0V 46890706 Ki > 2500 nM T66237 CIP1L7 46890707 Ki = 15 nM T66237 CKQ1Y0 46890708 Ki > 2500 nM T66237 C02IDZ 46890709 Ki = 600 nM T66237 CUWG39 46934434 IC50 > 100000 nM T66237 CI9J7N 47177173 Ki = 160 nM T66237 CO9JL6 47177176 Ki = 713 nM T66237 CMPE57 52941704 Ki > 10000 nM T66237 CBDS48 52949017 Ki > 10000 nM T66237 C01HUJ 53349364 Ki = 640 nM T66237 CK2Y5W 53349471 Ki = 98 nM T66237 C4TEY2 53358902 Ki > 10000 nM T66237 C63IVJ 53362154 EC50 = 3000 nM T66237 C21HMW 53362155 EC50 = 1698.24 nM T66237 CF60LM 53362156 EC50 = 1200 nM T66237 CGMY47 53362202 EC50 = 165.96 nM T66237 C9V8RI 53362203 EC50 > 10000 nM T66237 CAL1Y3 53362204 EC50 > 10000 nM T66237 C6N5EX 53362257 EC50 > 10000 nM T66237 CS40QD 53362258 EC50 > 10000 nM T66237 CFWL28 53362259 EC50 = 2600 nM T66237 CNDR76 53362310 EC50 > 10000 nM T66237 COUH09 53362311 EC50 > 10000 nM T66237 C1MU4B 53362312 EC50 > 10000 nM T66237 CLRT87 53362368 EC50 > 10000 nM T66237 CG8J6H 53362369 EC50 > 10000 nM T66237 CD1N3U 53362370 EC50 = 1600 nM T66237 CRY95P 53362428 EC50 = 720 nM T66237 C3TFA8 53362429 EC50 = 130 nM T66237 C4U1PT 53362430 EC50 = 138.04 nM T66237 C09KLV 53362488 EC50 = 257.04 nM T66237 CRX54F 53362489 EC50 = 186.21 nM T66237 C3KCI9 53362490 EC50 = 1100 nM T66237 CW32MV 53362546 EC50 > 10000 nM T66237 C5EG6T 53362547 EC50 = 5248.07 nM T66237 CUD9F0 53362548 EC50 = 1600 nM T66237 CVJ9U2 53362603 EC50 = 3700 nM T66237 CMY7V4 53362604 EC50 > 10000 nM T66237 CK9V1G 53362605 EC50 > 10000 nM T66237 CCRZ83 53362670 EC50 > 10000 nM T66237 CYK9B3 53362671 EC50 = 950 nM T66237 CCK0P6 53362672 EC50 > 10000 nM T66237 CYG85M 53362729 EC50 = 72.44 nM T66237 C1IBT7 53362730 EC50 > 10000 nM T66237 CI0F3Y 53362731 EC50 > 10000 nM T66237 C3XW1F 53362732 EC50 > 10000 nM T66237 CYTJ92 53362793 EC50 > 10000 nM T66237 CQ9CD8 53362794 EC50 > 10000 nM T66237 CAN2C1 53362795 EC50 > 10000 nM T66237 CO4UA0 53362796 EC50 = 389.05 nM T66237 C0NSZ5 53362797 EC50 > 10000 nM T66237 CFJO73 53362798 EC50 > 10000 nM T66237 C2RSW6 53362849 EC50 = 2500 nM T66237 C5K9YV 53362850 EC50 = 114.82 nM T66237 CB3AR7 53362851 EC50 = 200 nM T66237 C42SJF 53362852 EC50 > 10000 nM T66237 C8U6LX 53362853 EC50 > 10000 nM T66237 CH93SM 53362854 EC50 > 10000 nM T66237 C7RYJ0 53362909 EC50 = 330 nM T66237 CKV9D6 53362910 EC50 > 10000 nM T66237 CX9YM6 53362911 EC50 = 467.74 nM T66237 C76TQB 53362913 EC50 > 10000 nM T66237 C5XCD8 53362914 EC50 > 10000 nM T66237 C8N0TX 53362915 EC50 > 10000 nM T66237 CU9X3P 53362962 EC50 = 1200 nM T66237 C61CNE 53362963 EC50 = 1174.9 nM T66237 CF30CI 53362964 EC50 = 758.58 nM T66237 C6SB7W 53362965 EC50 = 970 nM T66237 C32FZM 53362966 EC50 > 10000 nM T66237 CJ06TA 53362967 EC50 > 10000 nM T66237 C6AN7Y 53363015 EC50 = 380 nM T66237 C52IOF 53363016 EC50 = 208.93 nM T66237 C1SHU3 53363017 EC50 = 2600 nM T66237 CNA2L1 53364234 Ki > 10000 nM T66237 C3L7RP 54580516 Ki > 1000 nM T66237 CX1H3Z 54580518 Ki > 1000 nM T66237 C7X4LI 54581307 Ki = 5200 nM T66237 CB5R2M 54581528 Ki > 1000 nM T66237 CR7GD2 54581529 Ki > 1000 nM T66237 CUW8C7 54581530 Ki > 1000 nM T66237 CD21EL 54581533 Ki > 1000 nM T66237 C0ZNY9 54582318 Ki = 31100 nM T66237 CQ7Z8U 54582526 Ki > 1000 nM T66237 C8UN6Y 54582950 IC50 = 8 nM T66237 C7MP0S 54584254 Ki >= 10000 nM T66237 C73IGF 54584265 Ki = 6714 nM T66237 CX5T1G 54584266 Ki = 4918 nM T66237 CIGN05 54584267 Ki = 22010 nM T66237 CC49GD 54584268 Ki = 45000 nM T66237 C9N2QH 54584476 Ki = 618 nM T66237 CD1A0H 54584477 Ki > 1000 nM T66237 CXPY04 54584478 Ki > 1000 nM T66237 CHR91Z 54585227 Ki = 1558 nM T66237 C8YD0H 54585429 Ki = 636 nM T66237 C5N7VS 54585431 Ki > 1000 nM T66237 C3MLH7 54586172 Ki >= 10000 nM T66237 CL79ME 54586390 Ki > 1000 nM T66237 C1N7LU 54586391 Ki > 1000 nM T66237 C60DIQ 54586392 Ki > 1000 nM T66237 CJ76VF 56657866 Ki > 10000 nM T66237 CQG9J6 56657868 Ki > 1000 nM T66237 C31CRV 56658409 EC50 = 1.4 nM T66237 C6T3VC 56658416 EC50 = 4.074 nM T66237 CJ5FQ4 56664848 Ki > 10000 nM T66237 C5V3ME 56664849 Ki > 10000 nM T66237 C3SYC9 56665377 EC50 = 9.12 nM T66237 CQN0G9 56668257 Ki > 10000 nM T66237 CU9DK4 56671721 Ki > 10000 nM T66237 CSL0C7 56671723 Ki > 10000 nM T66237 CK9L4C 56672570 EC50 = 31 nM T66237 C8GLI4 56675151 Ki > 10000 nM T66237 C05JPT 56678446 Ki = 930 nM T66237 CNZU65 56682530 Ki = 9.9 nM T66237 CAG71L 57391220 Ki > 10000 nM T66237 C26OTQ 57394727 Ki > 10000 nM T66237 CFM91W 57399933 Ki > 1000 nM T66237 CHG37B 57519947 Ki = 580 nM T66237 C0DB5C 57519948 Ki = 1800 nM T66237 C15NPY 57520031 Ki = 3700 nM T66237 CBTU57 67839485 Ki = 78 nM T66237 CD1IQ4 70685417 Ki = 1400 nM T66237 CCTZ13 70685423 Ki > 1000 nM T66237 CJM18X 71449932 Ki = 7.6 nM T66237 CUD97X 71451749 Ki = 26.1 nM T66237 C7BCA6 71451750 Ki = 187.7 nM T66237 CJGO63 71451752 Ki = 54.3 nM T66237 C8KO3M 71453576 Ki = 14.05 nM T66237 CG03VC 71455302 Ki = 1.93 nM T66237 C1WME0 71455306 Ki = 16.8 nM T66237 C0IZ5N 71457081 Ki = 5.69 nM T66237 CDU2C8 71460752 Ki = 25.3 nM T66237 CT8C1G 71460754 Ki = 12.7 nM T66237 CE2AI3 71462477 Ki = 0.83 nM T66237 C1Q6RX 71462479 Ki = 4 nM T66237 C8GV2J 71552165 IC50 = 10200 nM T66237 CR14LV 71552166 IC50 = 2000 nM T66237 CZG2O3 71720517 IC50 = 398.11 nM T66237 CPB34Y 73345487 Ki = 7.6 nM T66237 C8N1IS 73347164 Ki = 500000 nM T66237 C2Y4UX 73348432 Ki = 1.5 nM T66237 CKAC48 73348509 Ki = 4.8 nM T66237 COP37N 73348674 Ki = 1100000 nM T66237 C7GDP3 73350017 Ki = 24.1 nM T66237 CLC49J 73350187 Ki = 0.7 nM T66237 C8BRM6 73350188 Ki = 0.5 nM T66237 CS3GK0 73350258 Ki = 1000000 nM T66237 C8GQK9 73350823 Ki = 8700 nM T66237 CQ8UO2 73351518 Ki = 2.1 nM T66237 CY4IW8 73351519 Ki = 117 nM T66237 CG8AD1 73354500 Ki = 4416 nM T66237 CI8Z1B 73354581 Ki = 4.2 nM T66237 C5CDG2 73354746 Ki = 1500000 nM T66237 CQV35P 73356145 Ki = 3.6 nM T66237 CLMY01 76073634 EC50 = 330 nM T66237 C1YLV9 90468623 EC50 = 0.29 nM T66237 CGZ9F1 90469608 EC50 = 0.08 nM T66237 CLXN70 90469674 EC50 = 0.07 nM T66237 CRO49T 90469675 EC50 = 0.1 nM T66237 CSKZ30 90469676 EC50 = 0.39 nM T66237 C3FE9W 118476329 EC50 = 0.22 nM T66237 CGKN68 118476331 EC50 = 0.23 nM T66237 C2TGY7 118476332 EC50 = 0.35 nM T66237 C4HGR0 118476333 EC50 = 0.45 nM T66237 CL2UK1 118476335 EC50 = 0.22 nM T66237 C2G3FX 118476336 EC50 = 0.19 nM T66237 CR3O9G 118476337 EC50 = 0.1 nM T66237 C76ONJ 118476338 EC50 = 0.1 nM T66237 CC2UJ0 118476339 EC50 = 0.38 nM T66237 CTV5Z6 118476341 EC50 = 0.27 nM T66237 C81BRW 118476342 EC50 = 0.29 nM T66237 CRG4T1 118476343 EC50 = 0.12 nM T66237 C3YZ5M 118476344 EC50 = 0.32 nM T66237 C24TBU 118476346 EC50 = 0.26 nM T66237 CEP13D 118476347 EC50 = 0.22 nM T66237 C2RE7I 118476348 EC50 = 0.31 nM T66237 C5E0HL 118476355 EC50 = 0.25 nM T66237 CUMW51 118476356 EC50 = 0.21 nM T66237 C21GNB 118476357 EC50 = 0.1 nM T66237 C6KZH9 118476358 EC50 = 0.23 nM T66237 C69TMC 118476359 EC50 = 0.29 nM T66237 C5Z9SC 118476360 EC50 = 0.14 nM T66237 C36WLI 118476361 EC50 = 0.11 nM T66237 CX9YV2 118476362 EC50 = 0.21 nM T66237 C94FHB 118476365 EC50 = 0.19 nM T66237 CI1E7V 118476366 EC50 = 0.26 nM T66237 CY4WD9 118476367 EC50 = 0.33 nM T66237 CS7DP0 118476369 EC50 = 0.19 nM T66237 C7DAO4 118476383 EC50 = 0.31 nM T66237 C1KUY3 118476384 EC50 = 0.1 nM T66237 C5IFR0 118476385 EC50 = 0.27 nM T66237 C50MTE 118705579 Ki > 100000 nM T66237 C9HX7Z 118705580 Ki > 100000 nM T66237 CR3TZ0 118719818 EC50 = 4.2 nM T66237 CFG2V7 118719819 EC50 = 9.9 nM T66237 C4J6ZO 118719820 EC50 = 35 nM T66237 C9B2WS 118719821 EC50 = 1.8 nM T66237 CAFX95 118719822 EC50 = 690 nM T66237 CH74ZW 118719823 EC50 = 670 nM T66237 C7QI5K 118719824 EC50 = 40 nM T66237 CAP85S 118719825 EC50 = 450 nM T66237 CDR70N 118719826 EC50 = 450 nM T66237 CH0WU8 118719827 EC50 = 77 nM T66237 C1OMZ4 118719828 EC50 = 11 nM T66237 C72LOG 118719829 EC50 = 100 nM T66237 CD0P3Q 118719830 EC50 = 57 nM T66237 CAKC58 118719831 EC50 = 80 nM T66237 CIK48G 118719832 EC50 = 100 nM T66237 CDSK02 118719833 EC50 = 34 nM T66237 C9GSF2 118719834 EC50 = 68 nM T66237 CS89AW 118719835 EC50 = 30 nM T66237 CTWG46 118719836 EC50 = 84 nM T66237 COQ71F 118719837 EC50 = 82 nM T66237 CT3LR1 118719838 EC50 = 78 nM T66237 CX3R0J 118719839 EC50 = 180 nM T66237 CT3O7P 118719840 EC50 = 170 nM T66237 CW2F8P 118719841 EC50 = 380 nM T66237 CC9ZH4 118719842 EC50 = 66 nM T66237 C0LIH8 118719843 EC50 = 180 nM T66237 CYWM79 118719844 EC50 = 47 nM T66237 CGJ05D 118719845 EC50 = 57 nM T66237 CH3DE8 118720259 EC50 = 62 nM T66237 C3DLZ2 118720260 EC50 = 86 nM T66237 COD37S 118720261 EC50 = 230 nM T66237 CPNB13 118720262 EC50 = 1400 nM T66237 CW4Q3B 118720263 EC50 = 1400 nM T66237 CI1SA4 118720264 EC50 = 70 nM T66237 CX2K6O 118720265 EC50 = 52 nM T66237 COHG04 118720266 EC50 = 1100 nM T66237 CL2WY9 118720267 EC50 = 1300 nM T66237 C53KXO 118720268 EC50 = 500 nM T66237 CH2T3S 118720269 EC50 = 150 nM T66237 C7KCE4 118720270 EC50 = 2600 nM T66237 CEK5A6 118720271 EC50 = 73 nM T66237 C4OSR7 118720272 EC50 = 18 nM T66237 C2Z8IG 118720273 EC50 = 2000 nM T66237 C3SD1R 118720274 EC50 = 1200 nM T66237 CXGF75 118720275 EC50 = 110 nM T66237 CZ96MR 118720276 EC50 = 2100 nM T66237 CM1V0E 118720277 EC50 = 1000 nM T66237 CJB1T7 118720278 EC50 = 140 nM T66237 C4KHJ3 118720279 EC50 = 36 nM T66237 C85IJS 118720280 EC50 = 720 nM T66237 CMK0A4 118720281 EC50 = 210 nM T66237 C1KPF5 118720282 EC50 = 55 nM T66237 C9XE0M 118720283 EC50 = 1600 nM T66237 CXV09J 118720284 EC50 = 140 nM T66237 C2VF6Q 118720285 EC50 = 1400 nM T66237 CLE5W1 118720286 EC50 = 100 nM T66237 C8QYZ7 118720287 EC50 = 3000 nM T66237 CMC18U 118720288 EC50 = 250 nM T66237 CF1RM4 118720289 EC50 = 30 nM T66237 CTS3Q9 118720290 EC50 = 760 nM T66237 C3AOC2 118734334 Ki = 184 nM T66237 CT9D1K 118734335 Ki = 880 nM T66237 CBR9L6 118734336 Ki = 820 nM T66237 C7CNM8 132095331 EC50 = 0.2 nM T66237 C3NMS8 132822145 Ki = 170 nM T66237 CGI81M 132822146 Ki = 160 nM T66237 CC09BD 135192928 IC50 = 25665 nM T66237 CWQ30S 135192932 IC50 = 7320 nM T66237 CSQ0Y2 135192979 IC50 = 23047 nM T66237 CQI48P 135192983 IC50 = 32604 nM T66237 CS8A2H 135192997 IC50 = 21450 nM T66237 C86LKI 135413563 EC50 = 850 nM T66237 CM26GP 135506374 Ki >= 58.4 nM T66237 CT0A1P 135916059 Ki = 6.4 nM T66237 CHJ03T 135916060 Ki > 1000 nM T66237 CO6G5W 135916061 Ki > 1000 nM T66237 CAN9M3 135916069 Ki = 913 nM T66237 CH2L4N 135916070 Ki = 29 nM T66237 CO03UG 136961690 Ki = 913 nM T66237 C8R7MZ 137637867 Ki = 140 nM T66237 CW8AC7 137642420 Ki = 54 nM T66237 C8F4QJ 137648906 Ki = 1790 nM T66237 CO2S9U 137652605 Ki = 46 nM T66237 C7XTV3 145711714 EC50 = 41 nM T66237 C63UNT 145960494 EC50 = 3669 nM T66237 CIG1P6 145961670 Ki > 6000 nM T66237 C53JQB 145962220 EC50 = 3900 nM T66237 CRXH51 145963213 Ki > 6000 nM T66237 CY0FL4 145964296 Ki = 334 nM T66237 CS40EH 145965644 Ki < 10 nM T66237 CYSP85 145965794 Ki > 1000 nM T66237 CAHB80 145966126 Ki = 331 nM T66237 CYIE13 145970269 Ki > 1000 nM T66237 C3H7SY 145970757 Ki = 52 nM T66237 C43AQD 145971417 Ki > 1000 nM T66237 CJF16G 145972114 Ki > 1000 nM T66237 CPY61F 145972843 Ki > 1000 nM T66237 CI9G0B 145974527 Ki > 1000 nM T66237 CFQ05K 145974615 Ki < 10 nM T66237 CNF1J3 145974638 Ki = 1148 nM T66237 CVE64Z 145975166 Ki = 233 nM T66237 CJT06P 145976546 Ki = 100 nM T66237 CQ2IG7 145976595 EC50 = 4 nM T66237 CF14DJ 145976648 Ki = 121 nM T66237 CS5CD6 145977918 Ki > 1000 nM T66237 CT1PI4 145978570 Ki = 282 nM T66237 CTYI46 145978612 Ki > 1000 nM T66237 CC65HB 155513872 EC50 = 0.3 nM T66237 C8BKV3 155523986 EC50 = 0.08 nM T66237 C2IZ6F 155535667 EC50 = 0.17 nM T66237 CA6DC4 155542670 EC50 = 0.35 nM T66237 C7N8YM 155548766 EC50 = 1800 nM T66237 CP9TR0 10324985 Ki > 10000 nM T66237 D00NIT 9810140 Ki = 1.19 nM T66237 D00SGZ 9917025 Ki = 381 nM T66237 D01WHI 135413562 Ki = 0.67 nM T66237 D09RIE 44419028 Ki = 750 nM T66237 D0K5NV 44428109 Ki > 1000 nM T66237 D0L0RP 44428107 Ki > 1000 nM T66237 D0NC8V 6918854 Ki = 630.96 nM T66237 D0Q0OR 10461270 Ki > 1000 nM T66237 D0R7QC 44419039 Ki = 131 nM T66237 D0T4ML 5311202 Ki = 28000 nM T66237 D0W3IQ 44419025 Ki = 1.2 nM T66237 D0Y0SO 44419026 EC50 = 0.05 nM T66237 D0ZD0W 11366713 Ki = 1125 nM T22655 CZYM47 44287934 IC50 = 276000 nM T22655 CYW1J0 44318263 IC50 = 298000 nM T22655 C0X4WJ 44375633 IC50 = 219000 nM T22655 CB1I4O 44375924 IC50 > 500000 nM T22655 CD0X2A 44375925 IC50 = 126000 nM T33124 D07ACT 5479530 IC50 = 10000 nM T33124 D07MOX 439260 IC50 > 10000000 nM T33124 D0N0ES 938 IC50 = 1125000 nM T33124 D0X9RY 243 Ki = 2000 nM T33124 D01LAC 6437850 IC50 > 10000 nM T33124 CD5JX0 6097 IC50 > 100000 nM T33124 CFR5J9 6918 IC50 = 4400 nM T33124 CLE87P 7419 IC50 = 392000 nM T33124 CAZ4Q3 7436 IC50 > 1000000 nM T33124 CBHG51 9822 IC50 = 910 nM T33124 C18YBO 10009 IC50 > 10000000 nM T33124 CXD8L9 10700 IC50 = 7800 nM T33124 C5JS6C 11985 IC50 > 100000 nM T33124 CC4Q8S 12473 IC50 > 5000 nM T33124 C8S5IX 12476 IC50 = 3929000 nM T33124 C3MK6N 13401 IC50 = 2478000 nM T33124 CL70CJ 13650 Ki = 13 nM T33124 CG1LI5 14313 IC50 = 13140 nM T33124 C61YWO 16976 IC50 > 2500000 nM T33124 C1VBO0 18496 IC50 > 2500000 nM T33124 C03POM 28115 IC50 = 1150 nM T33124 CC2IU7 34037 IC50 > 10000000 nM T33124 CK4HU2 67658 IC50 = 1045000 nM T33124 CL89PK 72899 IC50 = 745 nM T33124 C9WSN7 72930 IC50 > 1000000 nM T33124 CU50OJ 73836 IC50 > 1000000 nM T33124 CA1EO9 74713 IC50 = 4600 nM T33124 CVI0R4 90269 IC50 > 100000 nM T33124 C1B3QA 94960 IC50 > 10000000 nM T33124 CS6Z8K 95048 IC50 = 720 nM T33124 CNOH14 97629 IC50 = 930 nM T33124 C2N7BJ 209069 IC50 = 220 nM T33124 CI98OR 210830 IC50 = 418 nM T33124 CDE95F 219248 IC50 = 10100 nM T33124 CXQ68R 225438 IC50 = 27000 nM T33124 C31RYP 234556 IC50 > 100000 nM T33124 C87CMX 235702 IC50 > 100000 nM T33124 CC24UA 278396 IC50 > 100000 nM T33124 CGOC06 279630 IC50 > 10000000 nM T33124 C2WQ9Y 305687 IC50 = 90 nM T33124 CI1KB2 319979 IC50 > 100000 nM T33124 C2ULI9 343030 IC50 > 5000 nM T33124 CFB6G2 349115 IC50 = 1300 nM T33124 CJR18X 351036 IC50 = 200 nM T33124 C2J1RE 351037 IC50 = 300 nM T33124 CU0EP6 351652 IC50 > 100000 nM T33124 CJ49VP 352208 IC50 = 253000 nM T33124 C0V8FN 354316 IC50 > 2500000 nM T33124 C49KEP 447315 IC50 > 10000000 nM T33124 CA92XL 458349 IC50 > 100000 nM T33124 C5K3ZJ 459531 IC50 > 5000000 nM T33124 CKXO12 568654 IC50 > 500000 nM T33124 CGZ01B 588192 IC50 > 100000 nM T33124 CK97ZC 637090 IC50 = 357000 nM T33124 CP58OT 637541 IC50 = 6269000 nM T33124 C0L9OX 735156 IC50 > 10000000 nM T33124 C79CFS 770980 Ki = 4590 nM T33124 COT5M0 773806 IC50 > 100000 nM T33124 CN5E4T 818159 IC50 = 4 nM T33124 CK19RN 818882 IC50 > 100000 nM T33124 CH0FY8 819049 IC50 = 36 nM T33124 CH7W9X 819050 IC50 > 100000 nM T33124 C10HYM 819556 IC50 > 100000 nM T33124 CV2OD0 820270 IC50 > 26200 nM T33124 CC6G4J 833670 IC50 = 199000 nM T33124 C6YKO9 2049051 IC50 = 21000 nM T33124 C0R1SD 2050103 IC50 > 10000000 nM T33124 CXL02M 2050132 IC50 > 100000 nM T33124 CRKD94 2062168 IC50 > 2500000 nM T33124 C9VNH4 2063443 IC50 = 900000 nM T33124 C0GJ3Y 2113906 IC50 = 7905000 nM T33124 CO1V8G 2512481 IC50 = 1104000 nM T33124 CJ70WI 2734324 IC50 > 100000 nM T33124 CU4Q0T 2769634 IC50 = 7300 nM T33124 C2J9ML 2781852 IC50 = 17.2 nM T33124 C9T1JS 2794584 IC50 = 1300 nM T33124 CPU87E 3264479 IC50 = 1200 nM T33124 C73BKE 3561548 IC50 = 38000 nM T33124 C51QOE 3686650 IC50 = 1832000 nM T33124 CC0LA2 4179726 IC50 > 10000000 nM T33124 C16EGI 4961254 Ki = 3.5 nM T33124 CW3T0B 5183334 IC50 > 100000 nM T33124 CU68IK 7141881 Ki = 31.7 nM T33124 CVSU04 9817917 IC50 > 100000 nM T33124 CN50HC 10261088 IC50 = 140 nM T33124 C7X8OB 10344711 IC50 > 100000 nM T33124 C5MV2C 10531257 IC50 > 100000 nM T33124 C9YA8W 10531300 IC50 = 50000 nM T33124 CRV54N 11171714 Ki = 1.7 nM T33124 COT47F 11299678 Ki = 7.2 nM T33124 CEK10J 11622394 IC50 = 269 nM T33124 C8WCD5 11804901 IC50 = 1400 nM T33124 CZ2H9W 12205754 IC50 = 600 nM T33124 C58UTM 12501973 IC50 = 200 nM T33124 C8GJ3Q 12527112 IC50 > 5000 nM T33124 CN43EO 12605957 IC50 = 360 nM T33124 C72TKZ 12703605 IC50 = 55000 nM T33124 CM34ZV 13271054 IC50 = 33 nM T33124 CY6CM5 13711789 IC50 > 100000 nM T33124 C39KXP 15187160 IC50 = 3260 nM T33124 CBC9U1 15219883 IC50 = 150 nM T33124 C1WTA4 15933663 IC50 > 5000 nM T33124 CPGJ74 16225169 IC50 = 1426 nM T33124 CX1V8D 18938079 IC50 > 100000 nM T33124 CJE9H3 18938081 IC50 = 8800 nM T33124 CJ92GZ 20317991 IC50 = 8 nM T33124 C7UE9X 20431233 IC50 = 155 nM T33124 C8XM6E 21194199 IC50 = 1340 nM T33124 CV96GA 21622350 IC50 = 16 nM T33124 CD4CO9 21625970 IC50 = 1130 nM T33124 CK0N1C 21626163 IC50 > 100000 nM T33124 COW47N 21661241 IC50 = 900 nM T33124 C5NC3Z 21931591 IC50 = 1440000 nM T33124 CXG78T 22556501 IC50 > 5000 nM T33124 CK36HZ 22556514 IC50 > 5000 nM T33124 C1E6MC 23354375 IC50 = 9 nM T33124 C40MNJ 23423218 IC50 = 343 nM T33124 CWP84K 24728218 IC50 = 120 nM T33124 CB0G4A 24815611 IC50 = 516 nM T33124 CMK53H 24815612 IC50 > 5000 nM T33124 CI35UR 24815613 IC50 = 4204 nM T33124 CSRP35 24972975 IC50 = 2750 nM T33124 C8IDU3 24978023 IC50 > 100000 nM T33124 CJ29DL 39733327 IC50 > 5000 nM T33124 C8TX1U 42281625 IC50 = 4000 nM T33124 CFYI84 42601491 IC50 > 30000 nM T33124 C8EK3R 42623200 IC50 = 2460 nM T33124 CJ4MD2 42623269 IC50 = 26130 nM T33124 CCAW14 42623272 IC50 = 74070 nM T33124 CV6X3I 44128604 IC50 = 3 nM T33124 C6UOJ1 44157408 IC50 = 4 nM T33124 CTZ25D 44157409 IC50 = 197 nM T33124 C53UPY 44157410 IC50 = 8 nM T33124 C9WI1U 44157412 IC50 = 32 nM T33124 C9XZV5 44157495 IC50 = 3 nM T33124 C67KDR 44157496 IC50 = 10 nM T33124 C0VG5Y 44157497 IC50 = 8 nM T33124 C15TSZ 44157498 IC50 = 38 nM T33124 C1KQA4 44157568 IC50 = 22600 nM T33124 CY3WA8 44157569 IC50 = 14400 nM T33124 CAS7T0 44157572 IC50 = 5 nM T33124 C3XUV4 44176138 IC50 = 100 nM T33124 CYO2V3 44176139 IC50 = 17300 nM T33124 CL6IU7 44576687 IC50 > 5000 nM T33124 C32UWQ 44576688 IC50 = 1153 nM T33124 CF20IT 44576689 IC50 > 5000 nM T33124 C60UWG 44576721 IC50 > 5000 nM T33124 CI1XM7 44576722 IC50 > 5000 nM T33124 CF46RK 44576723 IC50 > 5000 nM T33124 C9DRE2 44623061 Ki = 190 nM T33124 CB31ST 44726831 IC50 = 200 nM T33124 CC8U0N 45792205 IC50 = 347000 nM T33124 C1RGC0 49875138 IC50 > 100000 nM T33124 C4M2KG 59223400 IC50 = 20000 nM T33124 CI34QL 60143296 IC50 = 1.5 nM T33124 C0T4LE 71187181 IC50 = 3.9 nM T33124 CP0AZ1 71270044 IC50 = 1.4 nM T33124 CU2KV9 71270093 IC50 = 2.4 nM T33124 CQS64G 71270196 IC50 = 2.7 nM T33124 C1W2RE 71270198 IC50 = 3.8 nM T33124 CL6W3K 71270282 IC50 = 3.1 nM T33124 CI61AC 71270376 IC50 = 8.4 nM T33124 C7IU4W 71270397 IC50 = 2 nM T33124 C6XR9F 71270399 IC50 = 4.7 nM T33124 C4N5JH 71270479 IC50 = 4.9 nM T33124 CWV4I2 71270546 IC50 = 12 nM T33124 C0IS5L 71449458 IC50 = 20000 nM T33124 C8AZ1U 71449459 IC50 = 2000 nM T33124 C7XG8C 71449460 IC50 = 30000 nM T33124 CA6FM9 71449461 IC50 = 8000 nM T33124 C6SK0A 71449462 IC50 > 100000 nM T33124 C9YI1X 71451262 IC50 = 30000 nM T33124 CL2XW7 71451263 IC50 = 10000 nM T33124 CEQ5F1 71451264 IC50 = 50000 nM T33124 CMTJ62 71451276 IC50 = 3000 nM T33124 CACF59 71451277 IC50 = 40000 nM T33124 CPEM98 71453078 IC50 > 100000 nM T33124 CB8Y6P 71453079 IC50 = 30000 nM T33124 C8WE1K 71453080 IC50 = 9000 nM T33124 C38GXB 71454820 IC50 = 800 nM T33124 C38PBS 71454821 IC50 = 900 nM T33124 CNUJ38 71454822 IC50 = 70000 nM T33124 CL53DU 71456592 IC50 = 1000 nM T33124 C2YNK3 71456593 IC50 = 100 nM T33124 C3H6WR 71456594 IC50 = 20000 nM T33124 CG0X1K 71456595 IC50 = 4000 nM T33124 CMO34X 71456607 IC50 > 100000 nM T33124 CLXK57 71458455 IC50 = 100 nM T33124 CD7J0T 71458456 IC50 = 20000 nM T33124 C6QJ4A 71460302 IC50 = 70000 nM T33124 CBZ94K 71460303 IC50 = 80000 nM T33124 CUS05W 71460304 IC50 = 70 nM T33124 CU54RF 71460305 IC50 = 20000 nM T33124 C9LK8Q 71460306 IC50 = 80 nM T33124 CR30CZ 71462001 IC50 = 400 nM T33124 CCXS16 71505692 IC50 = 63 nM T33124 CVS4A1 71655533 IC50 = 13 nM T33124 CL03AI 71655534 IC50 = 120 nM T33124 C3TWJ4 71655535 IC50 = 300 nM T33124 C4KT0Z 71655536 IC50 = 670 nM T33124 CNT97G 71655604 IC50 = 2.2 nM T33124 CZ2Q4W 71655605 IC50 = 2.1 nM T33124 CP7SX0 71655670 IC50 = 13 nM T33124 CC04YH 71655735 IC50 = 10 nM T33124 CE34DT 71681571 IC50 = 500 nM T33124 COSM37 71681572 IC50 > 100000 nM T33124 C39ZSJ 71681730 IC50 = 800 nM T33124 C9CPV2 71681731 IC50 = 700 nM T33124 CZT49J 71681732 IC50 = 500 nM T33124 CL2EX8 71681733 IC50 = 3000 nM T33124 C7LA5I 71681734 IC50 = 900 nM T33124 CZ3SG0 71681735 IC50 = 800 nM T33124 C4OIY3 71681895 IC50 = 100 nM T33124 CA1QD2 71719322 IC50 > 1000000 nM T33124 CE9DN5 72793909 IC50 = 50 nM T33124 C0V8XQ 73295540 IC50 = 270 nM T33124 CKG17U 73295541 IC50 = 5100 nM T33124 CAS13P 73295701 IC50 = 40000 nM T33124 C0QM8G 73295702 IC50 = 1700 nM T33124 CR87BW 73295704 IC50 = 260 nM T33124 CA16QM 73295707 IC50 = 50 nM T33124 CR0OC5 73295872 IC50 = 80 nM T33124 C2FL4S 73295873 IC50 = 70 nM T33124 C1E7QX 73295874 IC50 = 90 nM T33124 CKQ3Z1 73295875 IC50 = 100 nM T33124 CPFB91 73295876 IC50 = 60 nM T33124 C5M3LR 73295877 IC50 = 40 nM T33124 CQT56C 73295878 IC50 = 80 nM T33124 CGD8X7 73295879 IC50 = 60 nM T33124 CQF14U 73295880 IC50 = 50 nM T33124 CXY98I 73296039 IC50 = 70 nM T33124 CC3OY6 73296040 IC50 = 120 nM T33124 C6JO4N 73296041 IC50 = 90 nM T33124 C9SP8Z 73296042 IC50 = 120 nM T33124 CGT0V3 73296043 IC50 = 160 nM T33124 CM49EJ 73296045 IC50 = 110 nM T33124 CDA1H9 73296046 IC50 = 220 nM T33124 CRWJ56 73296203 IC50 = 240 nM T33124 CO59BH 73296206 IC50 = 400 nM T33124 CJPM21 73296209 IC50 = 330 nM T33124 C42PEI 73296357 IC50 = 310 nM T33124 C9A4OJ 73296358 IC50 = 440 nM T33124 CUJ0M3 73296362 IC50 = 760 nM T33124 CRO37J 73296643 IC50 = 50 nM T33124 C28GVC 73296644 IC50 = 850 nM T33124 C5SY7R 73296645 IC50 = 470 nM T33124 CM67HU 90036033 IC50 = 2800 nM T33124 C0N6DR 90036293 IC50 = 100 nM T33124 C7BL0V 90036412 IC50 = 80 nM T33124 C3VZO0 90036575 IC50 = 100 nM T33124 CIV3X7 90036814 IC50 = 80 nM T33124 CRD5C3 110172411 IC50 > 100000 nM T33124 C9AGD1 119086959 IC50 = 230 nM T33124 C37OUM 119086960 IC50 = 210 nM T33124 CY7XA0 122189434 IC50 = 3300 nM T33124 CGC64V 122189435 IC50 = 80 nM T33124 C0GM6P 127048506 IC50 = 1380 nM T33124 CE48SG 127049189 IC50 = 340 nM T33124 C84UJE 130302628 IC50 > 10000 nM T33124 C6EO4Y 132091077 IC50 = 1300 nM T33124 CKG6Z5 135418577 IC50 > 5000000 nM T33124 CJN8Y5 135610212 IC50 > 500000 nM T33124 CN2Z8I 135894470 IC50 = 128 nM T33124 CZB3C9 135894471 IC50 = 784 nM T33124 C1QOJ9 135930270 IC50 > 50000 nM T33124 CJN0O2 135976840 IC50 > 5000 nM T33124 CV6TY5 137006778 IC50 = 60 nM T33124 CO25FI 137175021 IC50 = 30 nM T33124 CT16VM 137175066 IC50 = 30 nM T33124 CP7F4O 137175067 IC50 = 600 nM T33124 CWYD74 137175089 IC50 = 40000 nM T33124 CZ2R4V 137175100 IC50 = 100 nM T33124 CN02WV 137175101 IC50 = 90 nM T33124 C6IL7F 137175103 IC50 = 300 nM T33124 CEK6Q4 137175104 IC50 = 50 nM T33124 CL64XB 137175105 IC50 = 50 nM T33124 C20YPI 137175123 IC50 = 700 nM T33124 CAB72Q 137175141 IC50 = 70 nM T33124 CND13F 137175185 IC50 = 4000 nM T33124 CC2XQ7 137175265 IC50 = 200 nM T33124 CRMU97 137175266 IC50 = 60 nM T33124 C9P4YE 137459864 IC50 = 3981.07 nM T33124 CE9G2I 145967877 IC50 = 390 nM T33124 C8AO1L 145969548 IC50 = 490 nM T33124 CNG10S 145970871 IC50 = 5200 nM T33124 C8B6GK 145971079 IC50 = 6700 nM T33124 C1I6NU 145971095 IC50 = 8800 nM T33124 C93VJH 145991239 IC50 = 39000 nM T33124 CCN0P3 155545992 IC50 = 316.23 nM T33124 CM5YS3 155551104 Ki = 1000000 nM T33124 CA35OS 155560404 IC50 = 316.23 nM T33124 D05FMD 9447 IC50 = 3671000 nM T33124 D08JNG 867 IC50 > 10000000 nM T33124 D0ET2F 256208 IC50 = 1499000 nM T33124 D0F3CO 3840 IC50 = 2000 nM T33124 D0X0ER 344135 IC50 = 7870 nM T70490 D05UFG 10184653 IC50 > 10000 nM T70490 D0O8GK 71496458 IC50 = 32900 nM T70490 D0J6AU 10152654 IC50 > 10 nM T70490 D0YB3W 156414 IC50 = 2700 nM T70490 D0HM5J 118253852 IC50 = 3.981 nM T70490 C0XQP7 6917747 IC50 > 100000 nM T70490 CD54AH 6993099 Ki = 6200000 nM T70490 CBS6P7 8022437 IC50 = 11000 nM T70490 CXE30M 11334066 IC50 = 822 nM T70490 C9D6XI 11736400 IC50 = 172 nM T70490 C8D7BS 11771234 IC50 = 13 nM T70490 CN4IM8 11817961 IC50 = 96 nM T70490 C31MCN 13186896 IC50 > 100000 nM T70490 C6XPN4 16664855 IC50 = 18 nM T70490 CZ8DI1 23643986 IC50 = 70 nM T70490 CZPF48 23648277 IC50 > 10000 nM T70490 C31XJH 23648296 IC50 > 10000 nM T70490 CN0VA7 24822701 IC50 = 14 nM T70490 CQU38W 24900755 IC50 = 1727 nM T70490 C2S8VB 24901099 IC50 = 29 nM T70490 CIN28B 24901100 IC50 = 403 nM T70490 CD2EH0 24901101 IC50 = 191 nM T70490 CS7B3F 24901102 IC50 > 10000 nM T70490 CGI0U2 25023791 Ki = 10000 nM T70490 C3C8YJ 25174148 IC50 = 1.995 nM T70490 C5M1BT 25195691 IC50 = 158.49 nM T70490 CJ63ZU 42641779 IC50 = 158.49 nM T70490 CZM36T 42641892 IC50 = 39.81 nM T70490 CRYH80 42642459 IC50 = 1 nM T70490 C25ELB 44143088 IC50 = 34.67 nM T70490 CL0M7R 44143089 IC50 = 6918.31 nM T70490 C9QDC0 44143091 IC50 = 588.84 nM T70490 CDVC01 44268431 Ki = 180000 nM T70490 CK8EB3 44268436 Ki = 220000 nM T70490 CAPM01 44413250 IC50 = 6296 nM T70490 C7EKG5 44413251 IC50 = 9637 nM T70490 CCG5S4 44413390 IC50 = 137 nM T70490 CS6X7V 44426055 IC50 = 606 nM T70490 C8IB2W 44426056 IC50 > 100000 nM T70490 C9TFJ8 44464926 IC50 = 10 nM T70490 CYO0T1 44465454 IC50 = 7.943 nM T70490 CE83YL 44465721 IC50 < 0.3981 nM T70490 C6OC4Z 44607530 IC50 = 2100 nM T70490 CWMN69 46882864 IC50 = 2545 nM T70490 CQT8N7 46882865 IC50 = 271 nM T70490 CP47RN 46882866 IC50 = 8.2 nM T70490 C75BEM 46882867 IC50 = 1.7 nM T70490 C2PKZ9 46882868 IC50 = 880 nM T70490 CLV43E 46882869 IC50 = 336 nM T70490 CY2MQ1 46882870 IC50 = 2193 nM T70490 C0M4PL 46882914 IC50 = 250 nM T70490 CC94XY 46882915 IC50 = 67 nM T70490 C5X4SE 46883366 IC50 = 1230 nM T70490 CO5PD8 46883367 IC50 = 29 nM T70490 C9J4KG 46883368 IC50 = 5.8 nM T70490 CNA0W6 46883391 IC50 = 200 nM T70490 CW1RB0 46883392 IC50 = 630 nM T70490 CEB8W0 46883393 IC50 = 1580 nM T70490 CXST57 46883394 IC50 = 330 nM T70490 C7I6OU 46883395 IC50 = 17 nM T70490 CA6BD2 46883396 IC50 = 215 nM T70490 CP0V2B 46883425 IC50 = 3.8 nM T70490 C4WNV1 46883426 IC50 = 5.1 nM T70490 C16KZC 46883427 IC50 = 0.9 nM T70490 CQX57K 46883428 IC50 = 11 nM T70490 CQN34G 46883429 IC50 = 1 nM T70490 C0ZH2Y 46883430 IC50 = 0.7 nM T70490 C56QYZ 46883464 IC50 = 0.3 nM T70490 CEZ54V 46883465 IC50 > 3000 nM T70490 C2QM7R 46883466 IC50 = 12 nM T70490 CE80HK 46883467 IC50 = 1419 nM T70490 CHA61U 46883468 IC50 = 1832 nM T70490 CI2FX9 46883469 IC50 = 63 nM T70490 CM4O6Q 46883470 IC50 = 17 nM T70490 C68XTP 46883502 IC50 = 2502 nM T70490 CYN9C1 46883503 IC50 = 1081 nM T70490 C6FI5J 46883504 IC50 = 495 nM T70490 C7IOX5 46883505 IC50 = 133 nM T70490 C3I0FZ 46883506 IC50 > 10000 nM T70490 CUI91D 46905615 IC50 > 220 nM T70490 C9PAR7 46905616 IC50 = 790 nM T70490 CAFW31 49783666 IC50 = 0.7943 nM T70490 CN0B1V 49783830 IC50 = 0.2512 nM T70490 CNI1P6 49783903 IC50 = 0.7943 nM T70490 CGF65B 49783985 IC50 = 5.012 nM T70490 CI59MV 49797572 IC50 > 30000 nM T70490 C96CKU 49797573 IC50 = 14 nM T70490 C56OCA 53317528 IC50 = 1995.26 nM T70490 C7I9AO 53317529 IC50 > 25118.86 nM T70490 CM60RJ 53317530 IC50 > 25118.86 nM T70490 C5A6IH 53317737 IC50 = 1000 nM T70490 C6FEH9 53318816 IC50 > 25118.86 nM T70490 CJAX07 53318817 IC50 = 15848.93 nM T70490 CG5AP6 53318818 IC50 = 125.89 nM T70490 C0QV5D 53322753 IC50 = 2511.89 nM T70490 CHB96K 53324300 IC50 = 316.23 nM T70490 CR1L4Y 53325394 IC50 > 25118.86 nM T70490 CVU0J1 53326656 IC50 = 316.23 nM T70490 CFC91M 54769914 IC50 = 2.512 nM T70490 CF3XA9 57999656 IC50 = 158.49 nM T70490 CLA3R9 66645269 IC50 = 1.995 nM T70490 C62SML 90655967 IC50 = 25.12 nM T70490 CJ7LT3 90655968 IC50 = 12.59 nM T70490 CB61WC 90655969 IC50 = 3.981 nM T70490 CK5X2M 91826235 IC50 = 2.512 nM T70490 CGFK60 101201806 IC50 = 51 nM T70490 C8E4WS 102323332 IC50 = 1 nM T70490 CI9L7M 118253811 IC50 = 15.85 nM T70490 C3BAX2 118253818 IC50 = 6309.57 nM T70490 CL5C4K 118253824 IC50 = 7.943 nM T70490 CO53KU 118253851 IC50 = 12.59 nM T70490 C7YFQ0 118253855 IC50 = 15.85 nM T70490 CCH97D 118253857 IC50 = 31.62 nM T70490 C24IWU 118253859 IC50 = 39.81 nM T70490 CM63RL 118253870 IC50 = 12.59 nM T70490 CPBD92 118253877 IC50 = 63.1 nM T70490 CCG7Y6 118253883 IC50 = 5.012 nM T70490 CA72QZ 118253888 IC50 = 6.31 nM T70490 C63BSU 118260121 IC50 = 63.1 nM T70490 CTE34I 118720232 IC50 > 100000 nM T70490 CSD62B 118720233 IC50 > 100000 nM T70490 C9WF7Q 118720234 IC50 = 66000 nM T70490 C76HIO 118720235 IC50 = 18000 nM T70490 CAT1R6 118720236 IC50 > 100000 nM T70490 CGAF42 118720237 IC50 > 100000 nM T70490 CJ28KZ 118720238 IC50 > 100000 nM T70490 CPH2V9 118720239 IC50 > 100000 nM T70490 CQA83T 134131850 IC50 = 199.53 nM T70490 C7UNJ4 134132070 IC50 > 10000 nM T70490 CVAH73 134134180 IC50 = 398.11 nM T70490 CD6H8U 134134303 IC50 > 10000 nM T70490 C1RWN0 134134473 IC50 = 1000 nM T70490 CB93JM 134134976 IC50 = 1258.93 nM T70490 CZL0G9 134138927 IC50 = 158.49 nM T70490 C1W7EY 134140481 IC50 = 501.19 nM T70490 C6B5RW 134141023 IC50 = 39.81 nM T70490 CO9E0J 134145021 IC50 = 25.12 nM T70490 CI6FZ3 134147640 IC50 > 10000 nM T70490 C3DCQ9 134148503 IC50 = 501.19 nM T70490 C9OLA1 134148630 IC50 > 10000 nM T70490 C8SH1L 134154191 IC50 = 31.62 nM T70490 CTQY96 136117851 IC50 = 450 nM T70490 C3YHN7 146685679 IC50 = 32.3 nM T70490 C7TI5V 147202641 IC50 > 10000 nM T70490 CIK2C0 147243243 IC50 = 2150 nM T70490 C0JL2F 147323358 IC50 = 4 nM T70490 CUAY08 148018738 IC50 = 12.3 nM T70490 CH0NR2 148192765 IC50 > 10000 nM T70490 CT25HK 148412521 IC50 = 2.7 nM T70490 CWD7A1 148809433 IC50 = 2051 nM T70490 C0SW6H 148967294 IC50 = 6.5 nM T70490 CQK39B 149491764 IC50 = 3.9 nM T70490 C1ZX5D 149494192 IC50 = 1.9 nM T70490 CCU10W 149589615 IC50 = 505 nM T70490 CN6G2P 149839762 IC50 = 307.1 nM T70490 C4GCQ2 149933110 IC50 > 10000 nM T70490 C08LSG 150088178 IC50 = 154 nM T70490 CJZ3L2 150363449 IC50 = 783 nM T70490 C26MXO 150396261 IC50 = 1520 nM T70490 C3IPK7 150631495 IC50 = 271 nM T70490 CJ6A9B 150967523 IC50 = 221 nM T70490 CFXO59 151118910 IC50 = 499 nM T70490 CO6QT1 151217326 IC50 = 2.8 nM T70490 CMX4K7 151268438 IC50 = 4.9 nM T70490 CG6CN4 151286177 IC50 = 1605 nM T70490 C7RZO2 151821865 IC50 = 785 nM T70490 CDL4W5 151971947 IC50 = 1 nM T70490 CYN8L2 152157601 IC50 = 537 nM T70490 CJ2KV5 152225461 IC50 = 135.4 nM T70490 CKZ6H9 152242423 IC50 = 21.3 nM T70490 COE18M 152296790 IC50 = 175 nM T70490 CR0EQ1 152335936 IC50 = 835 nM T70490 C0IO7L 152457310 IC50 = 391.5 nM T70490 CZG2D5 152823047 IC50 = 2.3 nM T70490 CPF6I5 155518852 IC50 = 483 nM T70490 CQF3W2 155521718 IC50 > 10000 nM T70490 CXC8Q2 155522247 IC50 = 79.43 nM T70490 CMJO87 155528739 IC50 = 630.96 nM T70490 CY2HC7 155538869 IC50 = 6.31 nM T70490 CVGT48 155543410 IC50 = 0.3981 nM T70490 C2J5NY 155559747 IC50 = 50.12 nM T70490 CU67FS 155561515 IC50 = 50.12 nM T70490 CA8WQ7 155565392 IC50 = 1.585 nM T70490 D00FGA 73737 IC50 > 25118.86 nM T70490 D09FGQ 123985 IC50 = 770 nM T70490 D0IV5D 11241135 Ki = 2700 nM T70490 D0L9VP 5287864 IC50 = 2600 nM T70490 D0U4TA 44413276 IC50 = 4787 nM T70490 D0Y5IQ 44255320 IC50 = 10000 nM T73694 D09KTS 24821094 IC50 = 18 nM T73694 D0E6XR 3062316 IC50 = 5.3 nM T73694 D03HUX 49792852 IC50 > 10000 nM T73694 D0E3TC 44259 IC50 = 247 nM T73694 D0G5XV 135565884 IC50 = 33 nM T73694 D0O0LS 25141092 IC50 = 195 nM T73694 D03BNU 59604787 IC50 > 10000 nM T73694 D0T3ME 156422 IC50 > 30000 nM T73694 CJ2SQ9 683690 IC50 > 10000 nM T73694 C3PL7H 961174 IC50 > 10000 nM T73694 C9U7NK 1128774 IC50 = 520 nM T73694 C9RQC1 1521040 IC50 = 5600 nM T73694 CVZ37I 2351464 IC50 = 1900 nM T73694 CLH1T0 4376831 IC50 > 10000 nM T73694 CM5VN6 4600415 IC50 = 120 nM T73694 C9YK6Q 4603900 IC50 > 10000 nM T73694 C3LN1Y 5240683 IC50 = 5830 nM T73694 CY2UO9 5329275 IC50 = 2320 nM T73694 C9JT4S 11847343 IC50 > 10000 nM T73694 CA3I4T 24753787 IC50 > 50000 nM T73694 C7YG1N 24759534 IC50 = 1700 nM T73694 CQN3Z7 24825710 IC50 = 310 nM T73694 C1RP0I 25094211 IC50 = 500 nM T73694 CGT1W6 25144294 IC50 = 13 nM T73694 CNG96H 25210579 IC50 > 10000 nM T73694 C3VRO9 44557921 IC50 > 10000 nM T73694 CU3RF1 45139989 IC50 > 10000 nM T73694 CQGZ06 45139991 IC50 > 10000 nM T73694 CYT37A 46232443 IC50 > 50000 nM T73694 C48ZVW 46232555 IC50 = 32000 nM T73694 CS9B1U 46232556 IC50 > 50000 nM T73694 C7ON5A 46233287 IC50 > 10000 nM T73694 CF91RS 49843531 IC50 > 10000 nM T73694 CV8X0G 50924500 IC50 = 5.65 nM T73694 C2Y6QS 50938552 IC50 > 10000 nM T73694 C9NYP4 51036677 IC50 > 10000 nM T73694 C4WRY3 51037112 IC50 > 10000 nM T73694 CRI28Z 51037948 IC50 > 10000 nM T73694 C8NA4L 53384644 IC50 > 30000 nM T73694 CXA92G 53484170 IC50 = 10 nM T73694 C7UK2N 53484181 IC50 = 7 nM T73694 CKD9H6 53484182 IC50 = 9 nM T73694 CH05EO 53484183 IC50 = 7 nM T73694 CAR45T 53484184 IC50 = 6 nM T73694 CE1ZK6 54759168 IC50 > 10000 nM T73694 COM26L 56658690 IC50 = 177 nM T73694 C8DWL7 56658691 IC50 = 477 nM T73694 C8GJ9S 56658692 IC50 = 10 nM T73694 CK3A4Z 56658700 IC50 = 19 nM T73694 CRE75Z 56658839 IC50 = 75 nM T73694 C0JK4L 56658840 IC50 = 495 nM T73694 C1JD6Z 56658841 IC50 = 15 nM T73694 C98WRJ 56658842 IC50 = 38 nM T73694 C9R5IT 56658843 IC50 = 8 nM T73694 C2Z9YO 56662177 IC50 = 42 nM T73694 CR50XZ 56662178 IC50 = 11 nM T73694 C8NGC7 56662179 IC50 = 14 nM T73694 C3H0VQ 56662180 IC50 = 13 nM T73694 CWM35E 56662181 IC50 = 64 nM T73694 CB0VE5 56662182 IC50 = 38 nM T73694 CVBK03 56662332 IC50 = 16 nM T73694 CFW3I1 56665626 IC50 > 10000 nM T73694 C5XW3F 56665627 IC50 > 10000 nM T73694 CO96CB 56665628 IC50 = 51 nM T73694 CO51RL 56665629 IC50 = 97 nM T73694 CEI39Q 56665634 IC50 = 5 nM T73694 CG5K2Q 56665635 IC50 = 17 nM T73694 CVEM27 56665636 IC50 = 63 nM T73694 CDT3K4 56665637 IC50 = 156 nM T73694 CCD3U6 56665765 IC50 = 32 nM T73694 CVBF37 56665766 IC50 = 379 nM T73694 C9OB2T 56665767 IC50 = 72 nM T73694 CXO10E 56669082 IC50 = 1524 nM T73694 CF7K6A 56669083 IC50 = 319 nM T73694 CLE86K 56669084 IC50 = 391 nM T73694 C7JCP2 56669085 IC50 = 104 nM T73694 C9ZTL3 56669088 IC50 = 70 nM T73694 CC8F0R 56669218 IC50 = 254 nM T73694 CXW95K 56669219 IC50 = 23 nM T73694 C2GB4J 56672541 IC50 = 256 nM T73694 C5VS7B 56672542 IC50 = 12 nM T73694 C8R9TW 56672548 IC50 = 47 nM T73694 C0ROQ7 56672549 IC50 = 124 nM T73694 CI6K1R 56672550 IC50 = 156 nM T73694 CC5NQ4 56672551 IC50 = 7 nM T73694 CY0PA7 56672679 IC50 = 35 nM T73694 CP6AE8 56672680 IC50 = 68 nM T73694 C0GUO4 56672681 IC50 = 34 nM T73694 C25WIJ 56675923 IC50 = 355 nM T73694 CJA2N4 56675924 IC50 = 6 nM T73694 CWY32H 56676047 IC50 = 22 nM T73694 CR0CJ1 56679234 IC50 > 10000 nM T73694 CHB5T1 56679235 IC50 = 2643 nM T73694 CF3TD1 56679236 IC50 = 799 nM T73694 CF5YP1 56679374 IC50 = 10 nM T73694 C8QR1J 56679375 IC50 = 93 nM T73694 CLKP65 56682548 IC50 = 10 nM T73694 CW2YZ7 56682555 IC50 = 19 nM T73694 C1JWN7 56682556 IC50 = 7 nM T73694 CS9YF2 56682557 IC50 = 52 nM T73694 COM56E 56682674 IC50 = 109 nM T73694 C03OTV 56682675 IC50 = 3 nM T73694 CG2A4M 56682676 IC50 = 137 nM T73694 CPHX64 57325478 IC50 > 50000 nM T73694 CQ9BW4 57325479 IC50 > 50000 nM T73694 CVK0G4 58056356 IC50 > 50000 nM T73694 CXJ63M 59603829 IC50 > 100000 nM T73694 CQEU96 59603842 IC50 = 390 nM T73694 CV63UL 67240318 IC50 > 10000 nM T73694 C5DGR9 69036886 IC50 = 10000 nM T73694 COU73Y 71226944 IC50 = 60 nM T73694 C40JOZ 71235465 IC50 = 77 nM T73694 CCN01X 71547862 IC50 > 10000 nM T73694 CP5C7Y 76311266 IC50 = 5.7 nM T73694 C4GD6X 76311267 IC50 = 4.8 nM T73694 C9XZ0C 76311268 IC50 > 1000000 nM T73694 C29NOJ 76314857 IC50 = 9.2 nM T73694 CQT97B 76314858 IC50 > 1000000 nM T73694 CIV6B3 76318467 IC50 = 410 nM T73694 C4PRL2 76318468 IC50 = 55 nM T73694 CFTP19 76318469 IC50 = 26 nM T73694 CQ01AS 76318470 IC50 = 186 nM T73694 CV0C8D 76322137 IC50 = 13 nM T73694 C3QMZ9 76325759 IC50 = 21 nM T73694 C65WFX 76325760 IC50 = 4.7 nM T73694 CWG41I 76325761 IC50 = 479 nM T73694 CV9H0X 76329340 IC50 = 13 nM T73694 CJKG82 76329341 IC50 = 4.1 nM T73694 CCP9B2 76329342 IC50 > 1000000 nM T73694 CX8Q2U 76329343 IC50 > 1000000 nM T73694 CY1N5G 76332981 IC50 > 1000000 nM T73694 CXBD37 76332982 IC50 = 7.6 nM T73694 CJ2T9E 76332983 IC50 = 3.2 nM T73694 CL0UZ2 76332984 IC50 > 1000000 nM T73694 C9I2BO 76335834 IC50 = 5300 nM T73694 CPG3A5 86302574 IC50 > 30000 nM T73694 C1HW4B 89735655 IC50 > 100000 nM T73694 CY0UC4 90645194 IC50 > 10000 nM T73694 CTE8D6 90654489 IC50 = 4.41 nM T73694 C7OT8X 90654490 IC50 = 40.7 nM T73694 CTL9V6 90654491 IC50 = 43.5 nM T73694 CP8XL9 90654492 IC50 = 53.4 nM T73694 C34VGE 90654493 IC50 = 59.4 nM T73694 CA1KD0 90654494 IC50 = 64.5 nM T73694 C8T5IA 90654495 IC50 = 69.5 nM T73694 C5M3YN 90654496 IC50 = 75.6 nM T73694 CW4MA2 90654497 IC50 = 154 nM T73694 CYW6C8 90654498 IC50 = 155 nM T73694 C0IE3P 90654499 IC50 = 190 nM T73694 CY7BI2 118706214 IC50 > 10000 nM T73694 C1KQ4A 118714325 IC50 > 10000 nM T73694 C8VP5J 118714336 IC50 > 10000 nM T73694 CF80US 135406083 IC50 = 1680 nM T73694 CZFA70 135611366 IC50 = 933 nM T73694 CHA4N2 136013680 IC50 > 10 nM T73694 CSON28 136044162 IC50 = 58100 nM T73694 CQ8GK2 136044163 IC50 = 2540 nM T73694 C1XYU3 136044164 IC50 = 130 nM T73694 CIOP32 136044165 IC50 = 1290 nM T73694 C5PF2R 136044166 IC50 = 11750 nM T73694 CPMJ51 136044167 IC50 = 3900 nM T73694 CKQM03 136044169 IC50 = 1350 nM T73694 CV78CR 136044170 IC50 > 10000 nM T73694 C78HUT 136044171 IC50 = 1990 nM T73694 C1YUD0 136219394 IC50 > 10 nM T73694 CIU8W3 136254389 IC50 > 10 nM T73694 C2QV3C 136998781 IC50 = 360 nM T73694 C0NM9J 136998782 IC50 = 1300 nM T73694 CFE05J 136998783 IC50 = 200 nM T73694 CV53AZ 136998784 IC50 = 270 nM T73694 CXC69T 137321158 IC50 = 111 nM T73694 CZOD53 137633880 IC50 = 350 nM T73694 C7BJY5 137636807 IC50 = 113 nM T73694 CO89DX 137649100 IC50 = 48 nM T73694 CINE03 137652514 IC50 = 173 nM T73694 C28QUP 137652864 IC50 = 220.2 nM T73694 CF27EG 155511610 IC50 = 956 nM T73694 C0AN1O 155512752 IC50 = 626 nM T73694 C2MD1Q 155513187 IC50 > 10000 nM T73694 D08HFG 24809764 IC50 > 10000 nM T73694 D09HVH 135566652 IC50 > 10 nM T73694 D09PTP 57325421 IC50 = 73 nM T73694 D0IZ8M 56675928 IC50 = 2 nM T73694 D0N4LR 53469448 IC50 = 412 nM T39698 D03BNU 59604787 IC50 > 10000 nM T39698 CV63UL 67240318 IC50 > 10000 nM T39698 C2MD1Q 155513187 IC50 > 10000 nM T39698 D0C1DQ 6490494 IC50 = 7280 nM T84634 D0N0RU 82146 IC50 = 13500 nM T84634 D08UGX 60652 IC50 = 540 nM T84634 D0AA6Z 9799888 IC50 = 5.1 nM T84634 D09YUQ 127019 IC50 = 7800 nM T84634 C9LCD8 3823 IC50 = 12000 nM T84634 C3NS4E 132775 IC50 = 1300 nM T84634 CXQ40P 5862285 IC50 = 20000 nM T84634 C62RUG 9821132 IC50 = 10 nM T84634 CO39KV 9838239 IC50 = 39000 nM T84634 CI6V2U 9870337 IC50 = 10 nM T84634 C9VEF0 9949645 IC50 > 25000 nM T84634 CDLS47 10021552 IC50 = 4700 nM T84634 CKPQ58 11154980 IC50 = 25 nM T84634 C4GO0T 11231328 IC50 = 20000 nM T84634 CVO5A3 11235737 IC50 = 3.5 nM T84634 C3TF0M 11236452 IC50 = 24 nM T84634 CB7YS1 11315814 IC50 = 1.3 nM T84634 C9W0QH 11373414 IC50 = 5.2 nM T84634 C5VC8J 11406760 IC50 = 47 nM T84634 C5KMI6 11427427 IC50 = 10000 nM T84634 C0PWX2 11441615 IC50 = 35 nM T84634 C2KXN4 11475327 IC50 = 54 nM T84634 CYH36X 11493096 IC50 = 25000 nM T84634 C39PJT 11495962 IC50 = 16 nM T84634 CS0J3Q 11499978 IC50 = 25000 nM T84634 CEV5B3 11501485 IC50 = 73 nM T84634 CRV87M 11510548 IC50 = 7 nM T84634 CW51VQ 11523005 IC50 = 9000 nM T84634 C3QH2T 11558212 IC50 = 7000 nM T84634 CG24YV 11565407 IC50 = 5000 nM T84634 CVO62B 11582136 IC50 = 50000 nM T84634 CKW1Z2 11582790 IC50 = 77 nM T84634 C2H7WN 11590652 IC50 = 34 nM T84634 C1ZO5J 11595033 IC50 = 50000 nM T84634 C7S3EY 11618244 IC50 = 50000 nM T84634 C1MS3D 11623142 IC50 = 20000 nM T84634 C7OF9S 11633939 IC50 = 100 nM T84634 CMF5L2 11645016 IC50 = 50000 nM T84634 CFLM39 11652817 IC50 = 20000 nM T84634 CX4A9P 11659007 IC50 = 9000 nM T84634 CE4KR7 11688435 IC50 = 20000 nM T84634 C9UL1Q 11688471 IC50 = 10000 nM T84634 CM8R9J 11690073 IC50 = 6 nM T84634 CL5S9K 11719046 IC50 = 4.2 nM T84634 CI1P7M 11750760 IC50 = 12 nM T84634 C6TS4D 11773824 IC50 = 46 nM T84634 C98WNZ 14795724 IC50 = 2800 nM T84634 CYZ8E7 15950260 IC50 = 4500 nM T84634 CS8QM5 16039690 IC50 = 900 nM T84634 C1RV2O 23442837 IC50 = 4000 nM T84634 CVG5R8 25141344 IC50 = 500 nM T84634 CAWG69 44390123 IC50 = 37 nM T84634 CDZH20 44390134 IC50 = 50 nM T84634 CIOY83 44390142 IC50 = 14.4 nM T84634 CDQ90V 44390161 IC50 = 19 nM T84634 CS5NY3 44390206 IC50 = 48 nM T84634 CT5DF2 44390231 IC50 = 8 nM T84634 CH1QM4 44390265 IC50 = 335 nM T84634 C8V7OA 44410763 IC50 = 125 nM T84634 C0SXD3 44410799 IC50 = 20 nM T84634 C3PYC4 44410807 IC50 = 37 nM T84634 CB6H1M 44410808 IC50 = 34.7 nM T84634 CXM15V 44410812 IC50 = 583 nM T84634 CM4Z0T 44410814 IC50 = 1.6 nM T84634 CR4HX5 44410840 IC50 = 7.3 nM T84634 C73OZJ 44410841 IC50 = 11.2 nM T84634 C3NED2 44410860 IC50 = 46.7 nM T84634 C1EA6U 44410861 IC50 = 9 nM T84634 CU5E6C 44410862 IC50 = 5 nM T84634 CR5Y0N 44410871 IC50 = 3 nM T84634 C8IV5K 44410881 IC50 = 40 nM T84634 CBS59K 44411032 IC50 = 60 nM T84634 CRU1S5 44411036 IC50 = 34 nM T84634 C9J8MS 44411109 IC50 = 1.4 nM T84634 CFA64M 44411110 IC50 = 403 nM T84634 CD53XR 44411116 IC50 = 26 nM T84634 CINM87 44421467 IC50 = 800 nM T84634 CS9W1C 44421568 IC50 = 43000 nM T84634 CX2D7Y 44421596 IC50 = 4 nM T84634 C3J4IK 44445028 IC50 = 2200 nM T84634 CER28I 44547030 IC50 = 140 nM T84634 CCP59J 44547031 IC50 = 50 nM T84634 CYA5V4 44547032 IC50 > 1000 nM T84634 CECD12 44547033 IC50 = 0.3 nM T84634 C8V0RF 44547182 IC50 = 300 nM T84634 CGHQ08 44547183 IC50 = 0.35 nM T84634 C4OH1Q 44547184 IC50 = 290 nM T84634 C6K0OT 44547185 IC50 = 200 nM T84634 CZT18X 44547186 IC50 = 120 nM T84634 CYVB48 44547187 IC50 = 50 nM T84634 C0NPS7 44547331 IC50 = 12 nM T84634 C1O9MY 44547332 IC50 = 75 nM T84634 CB9NJ4 44547333 IC50 = 8 nM T84634 C02MSK 44547334 IC50 = 3 nM T84634 C8K2VD 44547335 IC50 = 40 nM T84634 CY6RM7 44547336 IC50 = 6 nM T84634 C4YST2 44547474 IC50 = 125 nM T84634 CJS5M2 44547475 IC50 = 400 nM T84634 CQZM23 44547476 IC50 = 140 nM T84634 CZ3YF8 44569168 IC50 > 50000 nM T84634 CTU37D 44569169 IC50 = 5000 nM T84634 COQ93E 44569170 IC50 = 35000 nM T84634 CQ4R9W 44569193 IC50 = 5000 nM T84634 CCW9S3 44569194 IC50 = 15000 nM T84634 CQ9V3E 44569195 IC50 = 1000 nM T84634 C5L3BW 44569196 IC50 = 2500 nM T84634 CHR3B7 44569222 IC50 = 1500 nM T84634 CQ6L0D 44569244 IC50 = 7000 nM T84634 C4X7SL 52951448 IC50 = 10 nM T84634 CG9N3R 52951561 IC50 = 8 nM T84634 CXKQ83 52951562 IC50 = 250 nM T84634 CWT95A 52951563 IC50 = 10 nM T84634 C2LB4Z 52951564 IC50 = 100 nM T84634 CY61IQ 52951683 IC50 = 40 nM T84634 CTH5P9 52951684 IC50 = 26 nM T84634 C2QIY0 52951823 IC50 > 1000 nM T84634 C2XV8F 54581365 IC50 = 3 nM T84634 C9PC5O 54758311 IC50 > 1000 nM T84634 C1MT9P 54758312 IC50 = 350 nM T84634 CK6E8U 71450543 IC50 > 1000 nM T84634 C0J7GV 71452887 IC50 = 450 nM T84634 CME8C6 71452888 IC50 = 9.4 nM T84634 C9RQK0 71452893 IC50 = 90 nM T84634 C6M4HK 71454655 IC50 = 100 nM T84634 C5F6TC 71454656 IC50 = 45 nM T84634 C7KL6A 71454657 IC50 = 5.7 nM T84634 CDJ7S2 71456381 IC50 = 16 nM T84634 CF8SN4 71457688 IC50 = 95 nM T84634 CO6VP9 71457689 IC50 = 200 nM T84634 C3C8IE 71458230 IC50 > 10 nM T84634 C7H3KI 71459597 IC50 = 85 nM T84634 CT83JM 71459598 IC50 = 250 nM T84634 C8WRL9 71459599 IC50 = 1000 nM T84634 C5RW7V 71460077 IC50 = 250 nM T84634 C1F5PV 71460078 IC50 = 700 nM T84634 CP4JI3 71460079 IC50 > 1000 nM T84634 C0PQ4J 71461338 IC50 = 1000 nM T84634 CH9E1A 71461802 IC50 = 14 nM T84634 CM4QL3 71461812 IC50 = 500 nM T84634 CH80VJ 71461813 IC50 = 6.7 nM T84634 CD81EJ 71463058 IC50 = 13 nM T84634 COJC78 71463059 IC50 > 1000 nM T84634 CEVW85 90659735 IC50 > 10000 nM T84634 CPW37E 117911702 IC50 > 5000 nM T84634 CH3L7C 117911715 IC50 > 5000 nM T84634 C87YKP 118727453 IC50 = 3040 nM T84634 C14EWO 118727454 IC50 = 3260 nM T84634 CYX1B9 118727455 IC50 = 2620 nM T84634 CU34VL 118727456 IC50 = 2810 nM T84634 CCI1P2 118727457 IC50 = 3020 nM T84634 CDV98T 118727458 IC50 = 5070 nM T84634 CSDL81 118727459 IC50 = 2830 nM T84634 CGQB23 118727460 IC50 = 3090 nM T84634 C05CPH 118727461 IC50 = 2730 nM T84634 C30IXV 118727462 IC50 = 4020 nM T84634 C2TV4J 118727463 IC50 = 3140 nM T84634 CUH6X7 118727464 IC50 = 2340 nM T84634 C89AOJ 118727465 IC50 = 3130 nM T84634 C9Y4FQ 118727466 IC50 = 5190 nM T84634 C06KVH 118727467 IC50 = 3350 nM T84634 C9YJ4H 118727468 IC50 = 3480 nM T84634 CMN01I 118727469 IC50 = 2070 nM T84634 C1PBO9 118727470 IC50 = 1360 nM T84634 C3X5GN 118727471 IC50 = 3220 nM T84634 C6G3NA 118727472 IC50 = 1870 nM T84634 CARH21 118727473 IC50 = 3210 nM T84634 CWI1Z8 121472067 IC50 = 270 nM T84634 CZP07X 121472068 IC50 = 10600 nM T84634 C4AD2S 121472069 IC50 > 5000 nM T84634 CT7YX5 121472072 IC50 = 240 nM T84634 CVX1Q8 121472075 IC50 = 340 nM T84634 CGK83X 121472076 IC50 = 1660 nM T84634 C9JBV4 121472081 IC50 > 5000 nM T84634 CJD30N 121472085 IC50 > 5000 nM T84634 CXAD12 121474361 IC50 = 110 nM T84634 C9JA6W 122190692 IC50 = 370 nM T84634 CCE2I8 122190693 IC50 = 650 nM T84634 CK2AJ7 122190694 IC50 = 790 nM T84634 CJQ2X5 122190695 IC50 = 540 nM T84634 C4SHV9 122190696 IC50 = 970 nM T84634 CCD9E8 122190697 IC50 = 220 nM T84634 C4WUJ1 122190698 IC50 = 600 nM T84634 C0Q7FL 122190699 IC50 = 620 nM T84634 CF0KD5 122190700 IC50 = 460 nM T84634 C09BCZ 122190701 IC50 = 1020 nM T84634 CI0MK6 122190702 IC50 = 410 nM T84634 CQ9L8H 122190703 IC50 = 740 nM T84634 CM82GH 122190704 IC50 = 840 nM T84634 CV9L3K 122190705 IC50 = 630 nM T84634 C0XY8O 122190706 IC50 = 1110 nM T84634 CWOC89 127031597 IC50 = 3500 nM T84634 D06RAM 10389639 IC50 = 60 nM T84634 D07VYX 10786043 IC50 = 200 nM T84634 D0F8JO 9951075 IC50 = 2.4 nM T84634 D0O6QU 2605 IC50 = 1630 nM T38875 D06ACW 6083 EC50 = 1519 nM T38875 D08UUL 46700756 IC50 = 101.62 nM T38875 CL7KB0 265479 EC50 = 1800 nM T38875 CKJP46 1825716 EC50 = 550 nM T38875 C1SVD2 2132479 IC50 = 2500 nM T38875 C18HKQ 9885748 IC50 = 46000 nM T38875 CVZ5X1 13042082 EC50 = 30000 nM T38875 CKV4G1 16079040 IC50 = 1500 nM T38875 C7YG1N 24759534 IC50 < 10 nM T38875 C4IY8M 45256689 EC50 = 8 nM T38875 C1R7WB 45256693 EC50 = 3 nM T38875 CEF64I 45273893 EC50 = 0.6 nM T38875 C2JHA7 45375932 EC50 = 13 nM T38875 C6EU8K 45375934 EC50 = 58 nM T38875 CHM6E5 45378798 EC50 = 300 nM T38875 C74OZB 46190967 EC50 = 97 nM T38875 CC17KH 46194961 EC50 = 1.2 nM T38875 CF38CI 51034107 EC50 = 1240 nM T38875 C4R8VQ 51034984 EC50 = 660 nM T38875 CMS4C2 53372240 EC50 = 4 nM T38875 C4W9XL 53372379 EC50 = 17 nM T38875 C1OGK6 54708532 EC50 = 800 nM T38875 CJ37NF 56591699 EC50 = 1490 nM T38875 C0PLM2 56591796 EC50 = 1240 nM T38875 CX93PS 56592835 EC50 = 1240 nM T38875 CT4E8R 56832546 IC50 = 26000 nM T38875 CXJ63M 59603829 IC50 = 26 nM T38875 CQEU96 59603842 IC50 = 4.6 nM T38875 CPD80M 60171744 EC50 = 1 nM T38875 C1Z3YP 60194103 EC50 = 630.96 nM T38875 CK6WO0 66552478 IC50 < 10000 nM T38875 CZ0V9E 67232851 EC50 = 870 nM T38875 C5DGR9 69036886 IC50 = 98 nM T38875 CXSI14 71718330 IC50 = 10000 nM T38875 C1TM3P 71720141 IC50 = 10000 nM T38875 COWG10 71748255 EC50 = 1.9 nM T38875 C95VYQ 71765798 EC50 = 57 nM T38875 CZ2NS1 71765801 EC50 = 80 nM T38875 C25TYS 71765951 EC50 = 43 nM T38875 C7Q5IH 71765955 EC50 = 1.3 nM T38875 CMZ4X2 71766100 EC50 = 47 nM T38875 C6PZY8 71767831 EC50 = 52 nM T38875 C19TPH 71767833 EC50 = 35 nM T38875 C6KQP7 71767991 EC50 = 7 nM T38875 C8Y2FX 86698571 EC50 = 53 nM T38875 CF0IS4 86698599 EC50 = 100 nM T38875 CWQA67 86698790 EC50 = 323 nM T38875 C6F3IK 86698802 EC50 = 8.3 nM T38875 C1HW4B 89735655 IC50 = 53 nM T38875 COSC89 89837093 EC50 = 24 nM T38875 CBY6J2 118053829 EC50 = 1 nM T38875 C24RMQ 118640135 EC50 = 11 nM T38875 C63DSU 118725336 EC50 = 1.1 nM T38875 CXG30B 118725337 EC50 = 184 nM T38875 CK1IS9 118725338 EC50 = 1840 nM T38875 CW1EO2 121396404 EC50 = 8 nM T38875 C9IMB0 121396405 EC50 = 59 nM T38875 CQMS08 121396411 EC50 = 38.1 nM T38875 CKCR81 121396412 EC50 = 76 nM T38875 C0U7DQ 134149170 EC50 = 3391 nM T38875 C3RWH7 134149412 EC50 = 3 nM T38875 C1S3NP 134150934 EC50 = 4 nM T38875 CUKT54 135398518 EC50 = 300 nM T38875 CJ1I5T 136183528 EC50 = 39.81 nM T38875 CY9G0L 137637206 EC50 = 62 nM T38875 CB1EZ5 137644835 EC50 = 1200 nM T38875 CVIM80 137651306 EC50 = 1600 nM T38875 CM5ZV6 137660838 EC50 = 270 nM T38875 CITW61 142771124 EC50 = 25118.86 nM T38875 CE0S8V 155532038 EC50 = 338.84 nM T38875 CG09DP 155548590 EC50 = 440 nM T38875 CZQM57 155554194 IC50 = 107.5 nM T59082 CTR94V 439281 Ki = 11000000 nM T59082 C68JEM 71623467 IC50 = 420000 nM T59082 CQ7H4I 76310828 IC50 = 40000 nM T59082 C4KA5F 76310829 IC50 = 7160000 nM T59082 CK7GZ9 76310830 IC50 = 5730000 nM T59082 C5UW2S 76310831 IC50 > 500000 nM T59082 CPNL61 76314448 IC50 = 4370000 nM T59082 C5XJR9 76314449 IC50 = 5150000 nM T59082 CWG83I 76318036 IC50 = 8790000 nM T59082 C5FNJ0 76318037 IC50 = 6490000 nM T59082 C7U3FD 76318038 IC50 > 500000 nM T59082 CNBD52 76318039 IC50 = 1010000 nM T59082 CWN58O 76321750 IC50 = 1020000 nM T59082 C6GCM4 76321751 IC50 = 13250000 nM T59082 CGE2N3 76321752 IC50 = 8640000 nM T59082 C06FQB 76325364 IC50 = 1340000 nM T59082 CNL49F 76325365 IC50 = 2410000 nM T59082 CUS61H 76325366 IC50 = 50000 nM T59082 CCY93X 76325367 IC50 > 500000 nM T59082 C5V3ZB 76325368 IC50 = 395000 nM T59082 CK6RA9 76332597 IC50 = 3890000 nM T59082 C7XGH3 76332598 IC50 = 14940000 nM T59082 C51OKC 86573947 IC50 = 310 nM T59082 CK5TZ1 122182803 IC50 = 34000 nM T59082 CRY0J4 122182804 IC50 = 1010000 nM T59082 CO4I6D 137631793 IC50 = 776000 nM T59082 CUH4X7 137638019 IC50 = 776000 nM T59082 CG9OE2 137653829 IC50 = 720000 nM T59082 C9B7YT 145979496 IC50 = 3200000 nM T59082 C2WPC9 145979996 IC50 = 100000 nM T59082 CRVW17 145981767 IC50 = 1400000 nM T59082 C4WM7S 145993839 IC50 = 450000 nM T59082 CAZ65D 155545302 IC50 = 481000 nM T59082 CU81IK 155569069 IC50 = 254000 nM T59082 D07LUR 185698 IC50 = 6400000 nM T59082 D0G6XS 17106 IC50 = 2950000 nM T59082 D0GS9E 18950 Ki = 13100000 nM T28132 C3G7VB 1234292 IC50 < 1000 nM T28132 CA2JU7 46911115 IC50 = 3981 nM T28132 C73VYX 46911116 IC50 = 200 nM T28132 CVD43F 56659471 IC50 = 79 nM T28132 C8SR2X 56659475 IC50 = 22 nM T28132 CNM68T 56662903 IC50 = 1071 nM T28132 CP2LW0 56662936 IC50 = 631 nM T28132 CX9FB0 56662937 IC50 = 6310 nM T28132 C8PQ0U 56666408 IC50 = 85 nM T28132 C7BQD3 56669824 IC50 = 126 nM T28132 CHAK86 56669827 IC50 = 1000 nM T28132 CU0KW5 56673309 IC50 = 398 nM T28132 CDX09S 56673310 IC50 = 1585 nM T28132 CK8U1S 56673311 IC50 = 1995 nM T28132 C0OYQ1 56676613 IC50 = 1000 nM T28132 C04IVB 56676641 IC50 = 316 nM T28132 CW37HG 56676642 IC50 = 631 nM T28132 CLF76V 56676643 IC50 = 794 nM T28132 C4QCS7 56676649 IC50 = 59 nM T28132 CZ98WA 56676650 IC50 = 537 nM T28132 C8QO3N 56679972 IC50 = 398 nM T28132 C4CY2J 56679973 IC50 = 1995 nM T28132 C7TR6Q 56679975 IC50 = 2131 nM T28132 CMWY31 56683305 IC50 = 10 nM T28132 CY5S9E 56683306 IC50 = 794 nM T28132 C3J2FI 56683309 IC50 = 158 nM T25847 D02EEJ 6479267 IC50 = 10.3 nM T25847 D0G7UX 5284373 IC50 = 8.78 nM T25847 C8RA6C 6476061 IC50 = 12.7 nM T25847 C31GDL 24814873 IC50 = 97.1 nM T25847 CWI47U 50899161 IC50 = 19.8 nM T25847 CHN71J 52940634 IC50 = 26.1 nM T25847 CQ83LE 52940669 IC50 = 25.2 nM T25847 C2H0IK 52940670 IC50 = 59.5 nM T25847 CPKZ45 52940671 IC50 = 28.9 nM T25847 C7MA9P 52941831 IC50 = 9.45 nM T25847 CH9QA8 52941859 IC50 = 17.2 nM T25847 C97YWD 52945243 IC50 = 30.5 nM T25847 CE05IO 52945473 IC50 = 151 nM T25847 C43LWJ 52945496 IC50 = 158 nM T25847 C3BCG7 52946681 IC50 = 66.8 nM T25847 CR63JF 52946682 IC50 = 20.6 nM T25847 CH8TZ9 52946683 IC50 = 79.7 nM T25847 C7KW3U 52947912 IC50 = 24.2 nM T25847 C4KAU1 52947949 IC50 = 1583 nM T25847 CGX04A 52947950 IC50 = 55.9 nM T25847 CDF54U 73333515 Ki = 35.2 nM T13057 D03DXN 66435 IC50 = 19900 nM T13057 D03SRY 259331 IC50 > 300000 nM T13057 D08QMX 5757 IC50 > 300000 nM T13057 D00MFW 92577 IC50 = 318 nM T13057 D0I2AN 86298439 IC50 = 200 nM T13057 CQ7GE6 20834 IC50 = 12640 nM T13057 CW68ZS 61672 IC50 = 24.1 ug.mL-1 T13057 CD6SZ4 69748 IC50 > 500000 nM T13057 CN2GL3 92576 IC50 = 300 nM T13057 C7KJ3B 114917 IC50 = 2570 nM T13057 C5X1YU 160254 IC50 = 22500 nM T13057 C4IRY2 164676 IC50 = 2590 nM T13057 CCEG90 259329 IC50 = 17100 nM T13057 CA8WX9 314313 IC50 = 39130 nM T13057 CM0IQ3 446665 IC50 = 91000 nM T13057 CELG48 998012 IC50 = 52070 nM T13057 CJ90PO 1159989 IC50 = 176000 nM T13057 CE3S9R 1820399 IC50 > 50000 nM T13057 CIV1E3 2775086 IC50 > 500000 nM T13057 CB7OS1 2964738 IC50 = 181000 nM T13057 CCHX35 3096032 IC50 = 42390 nM T13057 C2C5UW 3109390 Ki = 700 nM T13057 C3NL9W 3246406 IC50 = 4990 nM T13057 C9G0CA 3653077 IC50 = 29000 nM T13057 CGA0N7 3734796 IC50 > 60000 nM T13057 CTCI08 3784946 IC50 > 60000 nM T13057 CI7F3L 5098884 IC50 = 161 nM T13057 CSU5J3 5098885 IC50 = 97 nM T13057 CAW37X 5240714 IC50 > 60000 nM T13057 CPM09B 5327156 IC50 > 500000 nM T13057 C6XCJ8 6420094 IC50 = 1800 nM T13057 CH03PR 9866186 IC50 = 2100 nM T13057 C1ECT8 9867205 IC50 = 5000 nM T13057 CA75NG 9985013 IC50 = 60000 nM T13057 CYV93G 10172292 IC50 = 9000 nM T13057 CUV6M1 10198815 IC50 = 14000 nM T13057 C3A8JL 10256983 IC50 = 16000 nM T13057 CH45KB 10258785 IC50 = 10000 nM T13057 C9R7GJ 10260791 IC50 = 22000 nM T13057 C0D9QX 10372989 Ki > 30000 nM T13057 CT4H0O 11006141 IC50 = 32000 nM T13057 C2WP1J 11343454 IC50 = 2600 nM T13057 C1JAC5 11425923 IC50 = 3940 nM T13057 COIR53 11456678 IC50 = 1800 nM T13057 CM1XL8 11844603 IC50 > 100000 nM T13057 C75UVA 11844604 IC50 > 100000 nM T13057 C96HKI 11886168 IC50 = 2500 nM T13057 CPV08O 12658768 IC50 > 20000 nM T13057 CE8Y4G 13779016 IC50 = 201800 nM T13057 CWU92E 20866464 IC50 > 50000 nM T13057 CJKO23 20866499 IC50 > 50000 nM T13057 C12GAZ 21145366 Ki > 30000 nM T13057 C54IUM 21778115 IC50 > 50000 nM T13057 CWJ2N6 23577107 IC50 = 5370 nM T13057 CV07UA 23577108 IC50 = 19900 nM T13057 CS91QU 23577109 IC50 = 450 nM T13057 CJ7UP5 23577110 IC50 = 2270 nM T13057 CE9B6H 25014222 IC50 > 20000 nM T13057 CW69GS 25023777 IC50 = 4550 nM T13057 CSN1R4 25023778 IC50 = 1830 nM T13057 CW2H8L 25023779 IC50 = 2110 nM T13057 CR0E7L 25023780 IC50 = 500000 nM T13057 CZ4R5U 25023781 IC50 = 3910 nM T13057 C7KPR6 25023782 IC50 = 6400 nM T13057 CL41YO 25023783 IC50 = 10200 nM T13057 C40QFI 25147702 IC50 > 100000 nM T13057 C09KZA 25262525 IC50 = 36000 nM T13057 C4WM9S 25262527 Ki = 5200 nM T13057 C6ND7U 25640845 IC50 > 100000 nM T13057 C3P8XN 42644186 IC50 > 40000 nM T13057 C98IOF 42644187 IC50 > 40000 nM T13057 CL04IU 44156271 IC50 = 14000 nM T13057 C92TBJ 44324648 IC50 > 100000 nM T13057 CF3R6Y 44336593 Ki > 30000 nM T13057 CQ31LB 44356471 IC50 = 1540 nM T13057 CJUM36 44415112 IC50 > 100000 nM T13057 C46QTA 44423905 IC50 = 2200 nM T13057 C01HDT 44562085 IC50 = 2470 nM T13057 CT6WJ3 45271336 IC50 = 2900 nM T13057 CSA7P5 45378656 IC50 = 212000 nM T13057 C10PAG 45378788 IC50 = 7800 nM T13057 CY4FW6 45378789 IC50 = 10400 nM T13057 CPZW76 45378927 IC50 = 9100 nM T13057 CZW2K9 45378928 IC50 = 8000 nM T13057 CN3SI9 45378929 IC50 = 86000 nM T13057 CPY85V 45378930 IC50 = 9300 nM T13057 CY9O0P 45378931 IC50 = 12000 nM T13057 CYRC54 45482878 IC50 > 40000 nM T13057 CK98JB 45482885 IC50 > 40000 nM T13057 CQ5U3C 45482886 IC50 > 40000 nM T13057 C8Z7HX 45482894 IC50 > 40000 nM T13057 CCKE09 45482895 IC50 > 40000 nM T13057 CLGB06 46830252 IC50 > 10000000 nM T13057 C81CPM 46861833 IC50 = 15200 nM T13057 C0A9LD 46861834 IC50 = 12200 nM T13057 C83GCS 46882340 IC50 > 44000 nM T13057 CPEG29 46888174 IC50 = 9590 nM T13057 C2IU1Z 49796692 IC50 = 152000 nM T13057 C2NJ3B 51003508 IC50 = 14000 nM T13057 CMDB84 53316640 IC50 > 50000 nM T13057 C9GVU5 53317937 IC50 > 50000 nM T13057 CV4QD5 53317938 IC50 = 15700 nM T13057 CWT10N 53319270 IC50 > 50000 nM T13057 CRE6Y5 53319872 IC50 > 300000 nM T13057 CRC82E 53320578 IC50 > 50000 nM T13057 C8Y4KW 53320579 IC50 = 20600 nM T13057 CF35GK 53320580 IC50 = 17400 nM T13057 C04CYS 53320581 IC50 > 50000 nM T13057 CBI29Z 53321875 IC50 = 33300 nM T13057 C94WKB 53324565 IC50 > 50000 nM T13057 CNZY43 56589511 IC50 > 10000000 nM T13057 C53XYO 56589513 IC50 > 10000000 nM T13057 CHM5V3 56660070 IC50 > 120000 nM T13057 CHOF39 56670422 IC50 > 120000 nM T13057 CI9R8M 56670423 IC50 > 120000 nM T13057 CL3N0K 56673907 IC50 > 120000 nM T13057 CAL96I 56673908 IC50 > 120000 nM T13057 CEK3S2 56680547 IC50 > 120000 nM T13057 C72JTU 56681854 IC50 = 54300 nM T13057 CJ50EL 56681855 IC50 = 34500 nM T13057 CN3EW7 56683882 IC50 > 120000 nM T13057 C5CQY2 56683883 IC50 > 120000 nM T13057 CV4PW2 56683884 IC50 = 47600 nM T13057 CZP28F 57327772 IC50 = 20910 nM T13057 CG71TE 57380427 IC50 > 10000000 nM T13057 C4QJD7 57380429 IC50 > 10000000 nM T13057 CLTX25 57380431 IC50 > 10000000 nM T13057 CU94DW 57380433 IC50 = 191000 nM T13057 CCY75L 57380662 IC50 > 10000000 nM T13057 CE24LJ 57380664 IC50 = 210000 nM T13057 CWZ9E2 57380666 IC50 > 10000000 nM T13057 C9H7GI 57380668 IC50 > 10000000 nM T13057 CXW05S 57390693 IC50 > 10000000 nM T13057 CE57HQ 57395972 IC50 > 10000000 nM T13057 CGC16T 57397768 IC50 > 10000000 nM T13057 C18FTX 57397769 IC50 > 10000000 nM T13057 CQNG21 57397770 IC50 > 10000000 nM T13057 CX3A5R 57399431 IC50 > 10000000 nM T13057 CU5ND3 57514697 Ki = 6600 nM T13057 C4ZE0T 60142018 IC50 = 6900 nM T13057 COH1S4 60142154 IC50 = 7800 nM T13057 C49OYN 60142155 IC50 = 8000 nM T13057 CJ7AP3 67762287 IC50 > 20000 nM T13057 C2BT9H 70673568 IC50 = 2500 nM T13057 CUS3F6 70691280 IC50 > 100000 nM T13057 C3AJ7H 70981706 IC50 = 1800 nM T13057 CP4H6L 70981726 IC50 = 2200 nM T13057 C2KS7Y 70982811 IC50 = 1800 nM T13057 C7VES4 71449486 IC50 = 16670 nM T13057 CXI0F3 71561559 IC50 > 100000 nM T13057 CE0Y3O 71561685 IC50 = 4000 nM T13057 C3M4CF 71561686 IC50 = 3600 nM T13057 C82KCZ 71561687 IC50 = 2300 nM T13057 CDA8P2 71561688 IC50 = 38000 nM T13057 C87EXF 71561689 IC50 = 2830 nM T13057 CP9HX5 71561815 IC50 = 600 nM T13057 C9H5YS 71561816 IC50 = 5000 nM T13057 C61MWP 71561817 IC50 = 4500 nM T13057 C9GO5M 71561818 IC50 = 10900 nM T13057 CWA30F 71561819 IC50 = 4500 nM T13057 CBC4G0 71561820 IC50 = 5200 nM T13057 CPV8Y3 71561944 IC50 = 3600 nM T13057 CPWU40 71597177 IC50 = 31000 nM T13057 CT4MK9 71717989 IC50 = 30000 nM T13057 CCY15D 71734765 IC50 = 560 nM T13057 C6F1TD 72163289 IC50 = 13360 nM T13057 C0FWS2 72163422 IC50 = 13810 nM T13057 C2RNH4 72163424 IC50 = 21450 nM T13057 CNLB62 72163425 IC50 = 22290 nM T13057 CMC9L2 72190151 IC50 = 3400 nM T13057 CM1W6X 73352369 IC50 = 9200 nM T13057 C1DWU4 73353952 IC50 = 5300 nM T13057 C9UP3V 73353954 IC50 = 9890 nM T13057 CS5O4J 73355491 IC50 = 11660 nM T13057 CMDC47 73357035 IC50 = 6790 nM T13057 CY0K7L 73357036 IC50 = 10150 nM T13057 CH3V7I 76966642 IC50 = 12000 nM T13057 CERG27 86763337 IC50 = 4660 nM T13057 CGMI50 86763338 IC50 = 5420 nM T13057 CF05WT 86763339 IC50 = 220 nM T13057 CCFJ28 86763340 IC50 = 310 nM T13057 CD5W1T 86763452 IC50 = 420 nM T13057 CQE36J 86763453 IC50 = 630 nM T13057 CUX1G9 86764668 IC50 = 620 nM T13057 C2S3RG 86764669 IC50 = 660 nM T13057 C1W0XL 86764771 IC50 = 760 nM T13057 CW4A9E 86764772 IC50 = 770 nM T13057 CG5MU6 86764773 IC50 = 860 nM T13057 CNV49T 86764774 IC50 = 1050 nM T13057 CHD8N6 86764775 IC50 = 1200 nM T13057 CNW67M 86764883 IC50 = 1250 nM T13057 C0F7ES 86764884 IC50 = 1460 nM T13057 CWG7N1 86764885 IC50 = 1350 nM T13057 CGKE84 86764886 IC50 = 1490 nM T13057 C34KEY 86764887 IC50 = 1760 nM T13057 C6KM9C 86764996 IC50 = 1790 nM T13057 CP50RV 86764997 IC50 = 1840 nM T13057 C9KMS4 86764998 IC50 = 2310 nM T13057 CCR5O1 86764999 IC50 = 2390 nM T13057 CRU5W9 86765000 IC50 = 2730 nM T13057 CL4IN3 86766306 IC50 = 19740 nM T13057 CI8XJ4 90663933 IC50 > 5 nM T13057 CBK96X 90666455 IC50 > 20000 nM T13057 C61PBQ 90666456 IC50 > 20000 nM T13057 C40WCO 90666457 IC50 > 20000 nM T13057 C2ZGE9 90666458 IC50 > 20000 nM T13057 CG5TY1 90666459 IC50 > 20000 nM T13057 CWQN87 90666460 IC50 > 20000 nM T13057 CLU52N 90666461 IC50 = 19140 nM T13057 C0DW7A 90666462 IC50 > 20000 nM T13057 CXMC74 90666463 IC50 > 20000 nM T13057 CG36RV 91667928 IC50 = 14000 nM T13057 C19JKD 101884098 IC50 = 50000 nM T13057 CYW80L 102307785 IC50 = 2730 nM T13057 CL96MC 102532094 IC50 = 12500 nM T13057 C2BAM5 117803691 IC50 = 380 nM T13057 C6QM2W 118238298 IC50 = 70 nM T13057 CBEN51 118239663 IC50 = 300 nM T13057 C01WAG 118239984 IC50 = 1980 nM T13057 CPL19A 118247966 IC50 = 5700 nM T13057 CS41QV 118709487 IC50 = 14400 nM T13057 CL4IR5 118709488 IC50 = 370 nM T13057 CL8AK6 118709489 IC50 = 56000 nM T13057 CPDG83 118709490 IC50 = 2300 nM T13057 C8QWA7 118709491 IC50 = 3600 nM T13057 C8ISV6 118709492 IC50 = 5000 nM T13057 C6VAX0 118709493 IC50 = 4500 nM T13057 CLA0N9 118709494 IC50 = 5300 nM T13057 CR53LW 118709495 IC50 = 7200 nM T13057 C92GFL 118709496 IC50 = 8600 nM T13057 CP2V7L 118709497 IC50 = 10700 nM T13057 CIE91Q 118709498 IC50 > 20000 nM T13057 C3QK4Y 118709499 IC50 = 26000 nM T13057 CX2A8G 118722143 IC50 > 120000 nM T13057 CV5F0I 118722144 IC50 > 120000 nM T13057 C32ODE 118729111 IC50 = 6640 nM T13057 CTV62N 118729112 IC50 = 34620 nM T13057 CP9E4Q 118729113 IC50 = 18330 nM T13057 CS2XI7 118729114 IC50 = 10450 nM T13057 C3LN4T 118729115 IC50 = 8910 nM T13057 CF9KD7 118729116 IC50 = 9410 nM T13057 C27YKT 118729117 IC50 = 11460 nM T13057 C5FXC0 118729118 IC50 = 22250 nM T13057 C90UMX 118729119 IC50 = 24580 nM T13057 C0YGL1 118729120 IC50 = 13220 nM T13057 C4XZ2J 118729123 IC50 = 10870 nM T13057 C5GM1D 118729125 IC50 = 9690 nM T13057 CHF7U0 118729126 IC50 = 8250 nM T13057 C0M3VK 118729722 IC50 = 36800 nM T13057 CP4D5Q 118729725 IC50 = 33200 nM T13057 CWU09Y 118729729 IC50 = 31900 nM T13057 C0IJ2X 118737463 IC50 = 5400 nM T13057 C12OHP 122187565 Ki = 510 nM T13057 CXHR32 122187566 IC50 = 1400 nM T13057 C59OUG 122187567 IC50 = 2300 nM T13057 C2PVC5 122196288 IC50 = 11640 nM T13057 CUO46T 124140941 IC50 = 67 nM T13057 C04VCS 124140943 IC50 = 30 nM T13057 C0UAQ6 124147818 IC50 = 32 nM T13057 C8QAD1 124147824 IC50 = 37 nM T13057 C9SO3J 124147915 IC50 = 34 nM T13057 CS43YV 124147927 IC50 = 8 nM T13057 CZEC76 124147932 IC50 = 36 nM T13057 C5B4UL 124147957 IC50 = 50 nM T13057 C1KFO8 124147973 IC50 = 22 nM T13057 C70DOJ 124147979 IC50 = 27 nM T13057 C2VE5C 124148108 IC50 = 39 nM T13057 C3ER2Z 124148120 IC50 = 12 nM T13057 CH7OZ3 124148123 IC50 = 28 nM T13057 CFR2G7 124148125 IC50 = 260 nM T13057 CON3T6 124150358 IC50 = 105 nM T13057 CD5RM3 124150360 IC50 = 181 nM T13057 C25IJY 124150428 IC50 = 5 nM T13057 CHC02A 124150434 IC50 = 177 nM T13057 C04FYJ 124150499 IC50 = 23 nM T13057 C5H2QB 124150512 IC50 = 5 nM T13057 CD52ZW 124150523 IC50 = 429 nM T13057 CLJ36I 124150528 IC50 = 4 nM T13057 CE2W0X 124150540 IC50 = 31 nM T13057 C8N5JR 124150544 IC50 = 26 nM T13057 C9TB6E 124150550 IC50 = 28 nM T13057 C58EUN 124150620 IC50 = 10 nM T13057 C94XQA 124150663 IC50 = 12 nM T13057 C46PST 127024952 IC50 > 120000 nM T13057 CF05SB 127025572 IC50 > 120000 nM T13057 C0KDZ2 127025573 IC50 > 120000 nM T13057 CI0NR9 127025574 IC50 > 120000 nM T13057 C6RI3J 127025575 IC50 > 120000 nM T13057 C5Z4PH 127025576 IC50 > 120000 nM T13057 C94EIF 127025577 IC50 > 120000 nM T13057 CR87HW 127025578 IC50 > 120000 nM T13057 CM9CP5 127027398 IC50 > 120000 nM T13057 C2A4GS 127027399 IC50 > 120000 nM T13057 CYOQ30 127027703 IC50 > 120000 nM T13057 CX52UN 127027704 IC50 > 120000 nM T13057 C6TIJ1 127027705 IC50 > 120000 nM T13057 C6H9SE 127027706 IC50 > 120000 nM T13057 C2X4JK 127027707 IC50 > 120000 nM T13057 C6UR4C 127027724 IC50 > 120000 nM T13057 C0RQ1U 127027725 IC50 > 120000 nM T13057 C0K2UI 127028022 IC50 > 120000 nM T13057 C1WA5T 127028346 IC50 > 120000 nM T13057 CC8HW0 127028347 IC50 > 120000 nM T13057 C6T0DY 127028683 IC50 > 120000 nM T13057 CL6QV7 127028684 IC50 > 120000 nM T13057 CG68NT 127028685 IC50 > 120000 nM T13057 C3MCH5 127028686 IC50 > 120000 nM T13057 CIAX67 127050086 IC50 = 2160 nM T13057 CO8V1Q 134130829 IC50 > 20000 nM T13057 C9BH3S 134131790 IC50 = 114800 nM T13057 C3Q6HX 134132029 IC50 > 20000 nM T13057 COG29Y 134132248 IC50 = 6900 nM T13057 CXM14Y 134132344 IC50 > 20000 nM T13057 CY4N3A 134132971 IC50 = 12800 nM T13057 CJV5H9 134133280 IC50 = 8500 nM T13057 CQV2R8 134133435 IC50 = 9000 nM T13057 CIM15P 134134309 IC50 > 500000 nM T13057 CK1ED4 134137535 IC50 > 20000 nM T13057 CO69VN 134138834 IC50 = 392200 nM T13057 C9WV1I 134139428 IC50 > 20000 nM T13057 CCS63E 134140312 IC50 = 3500 nM T13057 CFVU60 134141414 IC50 = 20300 nM T13057 C4E0TR 134148396 IC50 > 20000 nM T13057 C9NU1K 134148434 IC50 = 136000 nM T13057 CRG1A0 134150611 IC50 > 20000 nM T13057 CR72FZ 134152023 IC50 = 19500 nM T13057 C1FGJ5 134152452 IC50 = 6700 nM T13057 CO24SI 134154614 IC50 = 19000 nM T13057 C5CU3J 134157618 IC50 > 20000 nM T13057 CN23HD 134157879 IC50 = 3200 nM T13057 CBD40I 135445085 Ki = 54500 nM T13057 CU29KR 135556239 IC50 = 1300 nM T13057 C72YQR 135647237 IC50 > 60000 nM T13057 CM40ZF 135656202 IC50 = 8658 nM T13057 CZLK13 135783298 Ki = 25600 nM T13057 CJC62N 135783299 Ki = 473600 nM T13057 CW61GO 135783300 Ki = 32300 nM T13057 C5OLC0 135783301 Ki = 388000 nM T13057 CI0ZD2 135783302 Ki = 11700 nM T13057 C7JY1E 135783303 Ki = 547500 nM T13057 CF1W0U 135783304 Ki = 1088200 nM T13057 CZC42X 135924009 IC50 = 4500 nM T13057 C5BL1Z 135924010 IC50 = 11900 nM T13057 C9UA3N 135924011 IC50 = 5000 nM T13057 C1V8JE 135924012 IC50 = 1300 nM T13057 C8HP1O 135924013 IC50 = 1400 nM T13057 CHUD85 135924014 IC50 = 5900 nM T13057 CTZ5K1 135924015 IC50 = 5500 nM T13057 CAF8B6 135924016 IC50 = 22900 nM T13057 CK4X8S 135924017 IC50 = 6300 nM T13057 CE1FB0 135924018 IC50 = 4800 nM T13057 C39EPD 135924019 IC50 = 8300 nM T13057 CEH2M5 135924020 IC50 = 10600 nM T13057 CN6I5O 135924021 IC50 = 15800 nM T13057 CKW8X5 135924023 IC50 = 22300 nM T13057 CO3EX1 135924024 IC50 = 4500 nM T13057 CBJ7F8 135924025 IC50 = 4400 nM T13057 C81SHP 135924026 IC50 = 3800 nM T13057 CI62JU 135924027 IC50 = 7400 nM T13057 CAL83P 135924028 IC50 = 1000 nM T13057 CJ14VX 135924029 IC50 = 5200 nM T13057 C5C4EP 135924030 IC50 = 800 nM T13057 C3OU8V 135924155 Ki = 18100 nM T13057 CE9O5C 135924156 Ki = 12900 nM T13057 CKMV15 135924157 Ki = 28700 nM T13057 CL32WR 135924158 Ki = 90800 nM T13057 CNF1P0 135924159 Ki = 103200 nM T13057 C0T8UJ 135924160 Ki = 11700 nM T13057 C76NSI 135924161 Ki = 16200 nM T13057 CZ0NP3 135924162 Ki = 22800 nM T13057 CQJ65M 135929084 Ki = 12300 nM T13057 C5QIK7 137174949 IC50 > 120000 nM T13057 CUF76K 137331590 IC50 = 46000 nM T13057 C9O8DG 137632552 IC50 = 4530 nM T13057 CPD4V1 137633197 IC50 = 1050 nM T13057 CA0G1S 137638114 IC50 = 14980 nM T13057 C7D4SW 137644380 IC50 = 940 nM T13057 CN1X0J 137651804 IC50 = 1700 nM T13057 CFV26J 137652273 IC50 = 180 nM T13057 CXQ40F 137653094 IC50 = 920 nM T13057 CQ7T4S 137653723 IC50 = 4700 nM T13057 CL4Z1R 137657281 IC50 = 1100 nM T13057 C4CY9T 137661102 IC50 = 15860 nM T13057 CRU6Z7 137796282 IC50 = 7670 nM T13057 C0WMZ4 139593950 IC50 > 36800 nM T13057 CTOP13 142357867 IC50 = 949 nM T13057 C6NQ9I 145720956 IC50 = 14000 nM T13057 C4DWG8 145950748 IC50 = 7760 nM T13057 CT6I5O 145961409 IC50 = 910 nM T13057 CX54KW 145965216 IC50 = 30620 nM T13057 C0UT4Z 145966104 IC50 = 15530 nM T13057 C5H4PZ 145966112 IC50 = 25800 nM T13057 C9ICD0 145966982 IC50 = 23920 nM T13057 C58OBV 145971193 IC50 = 1590 nM T13057 CUE85W 145971302 IC50 = 2110 nM T13057 C73LAX 145972390 IC50 = 26510 nM T13057 C4IKH8 145973652 IC50 = 29950 nM T13057 COKV83 145974730 IC50 = 10000 nM T13057 C82EIW 145976484 IC50 = 5810 nM T13057 C2OZ8G 145976572 IC50 = 13980 nM T13057 CC2YO9 155516358 IC50 = 4870 nM T13057 C3PVL6 155517759 IC50 = 7830 nM T13057 CGUP05 155517773 IC50 = 4260 nM T13057 C7L3BR 155518108 IC50 = 3290 nM T13057 C2LYI7 155518870 IC50 = 985 nM T13057 CDYT42 155519082 IC50 = 2280 nM T13057 CZ75SL 155521073 IC50 = 6930 nM T13057 C9SD1X 155522483 IC50 = 6544 nM T13057 C4IA1T 155522941 IC50 = 1300 nM T13057 CL3I5G 155526321 IC50 = 1573 nM T13057 CG5YL4 155527104 IC50 = 54000 nM T13057 CTB6J8 155531587 IC50 = 2180 nM T13057 C38HEA 155532611 IC50 = 3280 nM T13057 C3NIE0 155532810 IC50 = 277 nM T13057 CZ94EY 155534761 IC50 = 7743 nM T13057 CLZ31N 155536741 IC50 = 2670 nM T13057 CEPN70 155536960 IC50 = 7552 nM T13057 C8YO9Q 155537362 IC50 = 6 nM T13057 CQ63GA 155537698 IC50 = 3800 nM T13057 CRU6F2 155538623 IC50 = 5810 nM T13057 C3Y6ZF 155538861 IC50 > 38900 nM T13057 CLF25Z 155545436 IC50 = 1950 nM T13057 CL78UG 155545756 IC50 = 4600 nM T13057 CARH78 155548168 IC50 = 23500 nM T13057 C1N8YP 155548589 IC50 = 5650 nM T13057 CRH8J5 155548680 IC50 = 8110 nM T13057 C50TQN 155550512 IC50 = 3700 nM T13057 C3GD5P 155550890 IC50 = 1230 nM T13057 CN6G0X 155556117 IC50 = 55200 nM T13057 CA75HC 155556730 IC50 = 2940 nM T13057 CG3I4L 155557442 IC50 > 100000 nM T13057 C0XU6Z 155559063 IC50 = 22000 nM T13057 CJI90K 155559808 IC50 = 4110 nM T13057 C5E0GW 155560770 IC50 = 500 nM T13057 CD4E5F 155560948 IC50 = 99000 nM T13057 CR03FB 155562299 IC50 = 6500 nM T13057 CE74XH 155564341 IC50 = 3100 nM T13057 CL1S9J 155565716 IC50 = 7780 nM T13057 C7W5HT 155566457 IC50 > 37700 nM T13057 D01BZE 73659 IC50 > 40000 nM T13057 D0SJ2Q 10494 IC50 = 11620 nM T13057 D0U8IF 10114 IC50 = 9600 nM T18904 D00SUC 74766595 IC50 = 99 nM T18904 D03TPE 97394 IC50 = 1700 nM T18904 D05PXW 6451399 IC50 = 15300 nM T18904 D09NCT 53392492 IC50 = 3300 nM T18904 D0C8CI 45376513 IC50 = 14000 nM T18904 D0JQ9Z 575125 IC50 = 3300 nM T18904 D0WC4Z 45376646 IC50 = 13000 nM T18904 C25LHT 125134 IC50 = 72000 nM T18904 C76AMR 439391 IC50 = 24000 nM T18904 CT0H6S 439939 IC50 = 26000 nM T18904 C5K3ZJ 459531 IC50 = 501.19 nM T18904 C4C0EB 2816189 Ki = 3020 nM T18904 CW2JY7 5715254 Ki = 520 nM T18904 C2JW1I 6288112 Ki = 5500 nM T18904 CCYF63 9942424 IC50 = 1258.93 nM T18904 CW01ZQ 22581416 IC50 = 16700 nM T18904 CP65KR 22581444 IC50 = 13200 nM T18904 C75LNS 22581449 IC50 = 10900 nM T18904 CCAM68 22959876 IC50 = 14000 nM T18904 C9J8TY 25721068 IC50 = 25000 nM T18904 C7X3WA 28330466 IC50 > 100000 nM T18904 CB2H6R 44820611 IC50 = 33000 nM T18904 CP59WA 45376516 IC50 = 12000 nM T18904 C1WL2X 45376644 IC50 = 20000 nM T18904 C62OQG 45376778 IC50 = 10000 nM T18904 CGF78A 45376782 IC50 = 13000 nM T18904 C32PQB 45376911 IC50 = 17000 nM T18904 C7OJ5E 46899602 IC50 = 8700 nM T18904 CUMF70 46899605 IC50 = 6000 nM T18904 C2DBN5 46899607 IC50 = 800 nM T18904 C3G4QK 46899609 IC50 = 5500 nM T18904 C24GUR 46899759 IC50 = 11000 nM T18904 C6ZR3Y 46899761 IC50 = 22000 nM T18904 CLK96Z 46899763 IC50 = 8100 nM T18904 CBOM64 46899765 IC50 = 3200 nM T18904 C9ENX8 46899767 IC50 = 2000 nM T18904 CF2QL4 46899769 IC50 = 4400 nM T18904 CW10BJ 46901089 IC50 = 17000 nM T18904 C6Z1NU 46901246 IC50 = 120000 nM T18904 CC23YW 49847498 IC50 > 25000 nM T18904 CWP7L0 49848519 IC50 > 25000 nM T18904 CU8AX0 55281807 Ki = 1940 nM T18904 CVK29R 57386523 IC50 = 4690 nM T18904 C8VM6P 67283460 IC50 > 25000 nM T18904 CY21XA 70702122 IC50 = 34000 nM T18904 C5XA3R 71733941 IC50 = 23500 nM T18904 C4PW1L 71734037 IC50 = 2400 nM T18904 C14GIV 71735687 IC50 > 120000 nM T18904 CM02VN 71735839 IC50 = 100000 nM T18904 C4WS1H 71735840 IC50 = 65000 nM T18904 CT4YO5 71735841 IC50 > 120000 nM T18904 C2ZFM8 71735842 IC50 = 99000 nM T18904 CI5W0K 71735843 IC50 > 120000 nM T18904 CYF8O7 71767874 IC50 = 125.89 nM T18904 CFY18G 73333510 IC50 > 120000 nM T18904 CN5B4O 73352277 IC50 = 92000 nM T18904 CX23ZP 78426670 IC50 > 2500 nM T18904 CKXW73 78427224 IC50 > 2500 nM T18904 C63ATV 81750201 IC50 = 100 nM T18904 CS4Q1F 86268882 IC50 < 100 nM T18904 CRQ51Z 86346639 IC50 < 100 nM T18904 CW9F0K 89564218 IC50 < 1000 nM T18904 C83TUW 89825693 IC50 = 100 nM T18904 CFX8E0 90407594 IC50 > 10000 nM T18904 C2NA5I 91801131 IC50 = 3162.28 nM T18904 CP3DK0 96607511 IC50 = 200 nM T18904 C85UGZ 96608360 IC50 = 16500 nM T18904 CCZ4Q9 96617507 IC50 = 900 nM T18904 C10RDJ 101882871 IC50 = 15848.93 nM T18904 CY87WL 112499933 IC50 = 104200 nM T18904 C4FPD3 112726150 IC50 > 100000 nM T18904 C6YT2Q 118598059 IC50 = 104 nM T18904 C75JVN 122191451 IC50 = 19952.62 nM T18904 C59KNQ 122191457 IC50 = 79432.82 nM T18904 CM5X8J 122191459 IC50 = 63095.73 nM T18904 C7ASR0 122191460 IC50 > 100000 nM T18904 CRI6J4 122191461 IC50 > 100000 nM T18904 C75NJO 122191464 IC50 = 50118.72 nM T18904 C50VYK 122191465 IC50 = 39810.72 nM T18904 CSKY20 122191466 IC50 = 79432.82 nM T18904 CS3L8H 122191467 IC50 = 2511.89 nM T18904 CZ2NV1 122191468 IC50 = 5011.87 nM T18904 CYTW93 122191469 IC50 = 5011.87 nM T18904 CZV45H 122191470 IC50 > 100000 nM T18904 CZU02B 122191472 IC50 = 6309.57 nM T18904 CQ04FW 122191477 IC50 = 39810.72 nM T18904 CT6HG3 122191480 IC50 = 63095.73 nM T18904 C2OVF5 122196456 IC50 = 2800 nM T18904 C8ADX6 122196457 IC50 > 100000 nM T18904 C0BEV2 122196458 IC50 > 100000 nM T18904 C6TP8J 122196459 IC50 = 3700 nM T18904 CWJL93 122196460 IC50 > 100000 nM T18904 C6MN0G 122196461 IC50 > 100000 nM T18904 CO4Y6T 122196462 IC50 > 100000 nM T18904 C2QGM6 122196463 IC50 > 100000 nM T18904 C83MKU 122196464 IC50 > 100000 nM T18904 CY7E0F 122196465 IC50 > 100000 nM T18904 C5OS8R 122196466 IC50 > 100000 nM T18904 C17TXO 122196467 IC50 > 100000 nM T18904 CNO5H7 122196468 IC50 > 100000 nM T18904 CW7U8M 122196469 IC50 > 100000 nM T18904 CT9R8C 122196470 IC50 > 100000 nM T18904 CGB05N 122196471 IC50 = 19000 nM T18904 CJG7O8 122196472 IC50 = 6200 nM T18904 CGO9Q2 122196473 IC50 = 24000 nM T18904 CEVG21 122196474 IC50 = 1800 nM T18904 CP4T8R 122196475 IC50 = 82000 nM T18904 CFI31P 122196476 IC50 = 1600 nM T18904 CJF70B 122196477 IC50 = 5100 nM T18904 CL89QK 122196478 IC50 = 50000 nM T18904 C6H2YQ 122383780 EC50 = 9000 nM T18904 CT2UZ4 125377518 EC50 = 3800 nM T18904 CF7KD3 127030402 Ki = 420 nM T18904 C63NWD 127030711 IC50 < 1000 nM T18904 CXF0U5 127030712 IC50 < 1000 nM T18904 CN16WB 127030937 IC50 = 1000 nM T18904 C2FPM6 127031758 IC50 = 30600 nM T18904 C7W8TS 127031759 IC50 = 300 nM T18904 CMJE83 127031760 IC50 = 950 nM T18904 CDC17F 127032730 IC50 = 100 nM T18904 CL38FP 127033048 IC50 = 100 nM T18904 CEV3A1 133053816 IC50 = 230000 nM T18904 C2Z6CV 135567105 IC50 = 11500 nM T18904 CIW61V 135567106 IC50 = 1700 nM T18904 CNZ8K9 135567107 IC50 = 8000 nM T18904 CL9ZD4 135567108 IC50 = 900 nM T18904 CJM4Z2 135567109 IC50 = 4100 nM T18904 CDY98J 135567110 IC50 = 138 nM T18904 C1VAI3 135567112 IC50 = 126 nM T18904 CWI0N7 135567114 IC50 = 16700 nM T18904 C8LFY7 135567115 IC50 = 80 nM T18904 C5E0ZN 135567116 IC50 = 15600 nM T18904 CO1F4A 135567128 IC50 = 630.96 nM T18904 CWCY64 136048725 IC50 = 21800 nM T18904 CE1SW8 136053677 IC50 = 630.96 nM T18904 CMW30T 136053680 IC50 = 794.33 nM T18904 C6IJ5M 136053683 IC50 = 1584.89 nM T18904 CNY5T7 136053684 IC50 = 398.11 nM T18904 C2V6MX 136644692 IC50 > 100000 nM T18904 CF5XJ1 137146154 IC50 = 6900 nM T18904 CK8DR7 137174994 IC50 = 1400 nM T18904 CA6DH2 137174995 IC50 = 1800 nM T18904 CLDH80 137174999 IC50 = 390 nM T18904 CR37AY 137175000 IC50 = 660 nM T18904 C1J3YB 137175001 IC50 = 600 nM T18904 CGAS95 137175002 IC50 = 880 nM T18904 CS5C6F 137175084 IC50 = 42800 nM T18904 C7PZ2T 137175085 IC50 = 6100 nM T18904 C1B5CK 137175086 IC50 = 13100 nM T18904 CWV4Y6 137175087 IC50 > 100000 nM T18904 C9XOV5 137175088 IC50 = 58600 nM T18904 C34LUV 137175094 Ki = 3 nM T18904 CSWN28 137175120 IC50 = 138 nM T18904 C23GYQ 137175121 IC50 = 110 nM T18904 C8Y2PR 137175122 IC50 = 128 nM T18904 C7GUC3 137175140 IC50 = 136 nM T18904 CBD1Q8 137175175 IC50 = 600 nM T18904 CEL6B1 137175176 IC50 = 770 nM T18904 C7SC6T 137175177 IC50 = 175 nM T18904 CPU73A 137175178 IC50 = 123 nM T18904 CFJ76N 137175179 IC50 = 411 nM T18904 CA89LW 137175180 IC50 = 456 nM T18904 C5GV3Q 137175209 IC50 = 145 nM T18904 C93YUK 137175210 IC50 = 143 nM T18904 CB2XV7 137175225 IC50 > 100000 nM T18904 C0XN8Y 137175239 IC50 = 9800 nM T18904 CI4D3P 137175249 IC50 = 181 nM T18904 CTVD83 137175250 IC50 = 147 nM T18904 C80LCT 137175251 IC50 = 158 nM T18904 CKQ1I2 137175252 IC50 = 144 nM T18904 C1YGB9 137175253 IC50 = 540 nM T18904 C5OZR6 137175260 IC50 = 109 nM T18904 CIKW02 137175261 IC50 = 118 nM T18904 C91JZQ 137321153 IC50 = 5300 nM T18904 C0D7SY 137349487 IC50 = 290000 nM T18904 C7J1RC 138393333 IC50 = 2060 nM T18904 CYG29R 138393334 Ki = 4 nM T18904 CNG82D 138393336 Ki = 4 nM T18904 CPFZ83 138393339 IC50 = 613 nM T18904 CC6SU2 138393341 Ki = 5 nM T18904 CXV31U 138753208 IC50 = 131 nM T18904 C41KVR 138753209 IC50 = 77 nM T18904 CIQJ26 138753211 Ki = 2 nM T18904 CARJ34 138753212 Ki = 26 nM T18904 C6LWR4 145963760 IC50 = 81 nM T18904 C0RPS4 145964567 IC50 = 41 nM T18904 CONJ19 145965089 EC50 = 105000 nM T18904 C3U8OD 145966600 IC50 = 615 nM T18904 CM9X8H 145967298 IC50 = 11 nM T18904 C9U5TQ 145967792 IC50 = 23 nM T18904 CB97SG 145968018 IC50 = 34 nM T18904 CT5MO6 145971004 IC50 = 82 nM T18904 CK9V5O 145972063 IC50 = 17 nM T18904 CX4W7P 145975124 EC50 = 1216000 nM T18904 CC8KI6 145976146 IC50 = 31 nM T18904 CKU0D3 145976400 IC50 = 208 nM T18904 CQ4E0O 145977225 IC50 = 269 nM T18904 CIQ6Y7 145977327 IC50 = 6 nM T18904 C5TBS2 145977546 IC50 = 41 nM T18904 CL2FR4 145978064 IC50 = 43 nM T18904 C8OL2Q 145978411 IC50 = 373 nM T18904 CA8UD0 145978535 IC50 = 15 nM T18904 C0GX1R 145985174 IC50 = 4200 nM T18904 C0UEA8 145992575 IC50 = 2200 nM T18904 CEQD63 155510449 IC50 = 246 nM T18904 CCB54Y 155510907 IC50 = 143 nM T18904 CAMR98 155512849 IC50 = 68 nM T18904 C9TWS3 155514456 IC50 = 59 nM T18904 C7XNM9 155518054 IC50 = 1060 nM T18904 C4M1EO 155519111 Ki = 4 nM T18904 CRT5Z2 155525082 IC50 = 848 nM T18904 CMB9N3 155530704 IC50 = 184 nM T18904 C2HN9G 155536799 IC50 = 282 nM T18904 C7VX3Y 155538517 IC50 = 178 nM T18904 C6YJ5R 155539215 IC50 > 25000 nM T18904 CP8K5E 155540290 IC50 = 71 nM T18904 C7LFH3 155540572 IC50 = 2410 nM T18904 COL30E 155540589 IC50 > 25000 nM T18904 CTF1K9 155542268 IC50 = 141 nM T18904 C7EG9J 155543678 IC50 = 188 nM T18904 C3M0TR 155546359 IC50 = 756 nM T18904 CTU53I 155547264 IC50 = 42 nM T18904 C5MFJ8 155548449 IC50 = 12350 nM T18904 CIM7D4 155548682 IC50 = 25000 nM T18904 C1CNK5 155549007 IC50 = 212 nM T18904 CX9OP1 155550806 IC50 = 259 nM T18904 CN7H9B 155554391 IC50 > 25000 nM T18904 C48ANL 155557731 IC50 = 88 nM T18904 C4MU5J 155558505 IC50 = 693 nM T18904 CTDM51 155558717 IC50 = 136 nM T18904 C0GU8Y 155559177 IC50 > 25000 nM T18904 CPOM30 155560356 Ki = 3 nM T18904 CGU0A2 155563031 IC50 > 25000 nM T18904 CA9T8I 155563296 IC50 = 218 nM T18904 C32NYC 155565735 IC50 > 25000 nM T18904 CGCN43 155567831 IC50 = 103 nM T18904 C3SQ4A 155569285 IC50 = 83 nM T18904 D07IOY 10365 IC50 = 4200 nM T18904 D08IZY 3080614 IC50 = 250000 nM T18904 D0B2WZ 15331 IC50 > 3300000 nM T18904 D0P7MU 4119262 IC50 = 20900 nM T18904 D0S3DD 56963315 IC50 = 400000 nM T18904 D0X5US 459617 IC50 = 1700 nM T22717 CU7X3G 2384714 IC50 > 5000 nM T22717 CRCA04 13590499 IC50 = 1700 nM T22717 CJ8YF2 13590558 IC50 > 5000 nM T22717 C1KN9T 24938152 IC50 = 310 nM T22717 C9EZ0X 25016113 IC50 = 830 nM T22717 C1WNJ5 25016370 IC50 = 520 nM T22717 CW7ZY1 25016377 IC50 = 720 nM T22717 CO7TN0 25016625 IC50 = 330 nM T22717 C1Q7XM 25016626 IC50 = 400 nM T22717 C4RA5E 25016628 IC50 = 150 nM T22717 C8VWT2 25016629 IC50 > 5000 nM T22717 CHC32Q 25016630 IC50 = 560 nM T22717 C6MOR1 25016631 IC50 = 1760 nM T22717 C0KR6F 25016883 IC50 = 260 nM T22717 C1G2EV 25016886 IC50 = 270 nM T22717 C87SMQ 25016887 IC50 = 210 nM T22717 CM19XI 25016888 IC50 > 5000 nM T22717 CL8S6A 25016889 IC50 = 2770 nM T22717 C4ML3F 25095022 IC50 = 660 nM T22717 C6M2FV 25095025 IC50 > 5000 nM T22717 CXGU79 25096820 IC50 = 150 nM T22717 CD7V1J 25097072 IC50 = 320 nM T22717 C3KGR7 25097315 IC50 = 2190 nM T22717 CAC4H7 25097316 IC50 = 430 nM T22717 CH8DY0 25097317 IC50 = 520 nM T22717 C95MYB 25097319 IC50 = 1040 nM T22717 C4GFB3 25097320 IC50 = 390 nM T22717 CJA2M5 25097322 IC50 > 5000 nM T22717 C37PQX 25097579 IC50 = 2820 nM T22717 C7N0JG 25097580 IC50 > 5000 nM T22717 CML61T 25097581 IC50 = 360 nM T22717 C1MQ5P 25097582 IC50 = 910 nM T22717 CFQY57 25097583 IC50 = 770 nM T22717 C9NKV4 25098135 IC50 = 640 nM T22717 C04ZFM 25098136 IC50 = 1220 nM T22717 CF01QP 25098137 IC50 = 710 nM T22717 CA0BL7 25098138 IC50 = 1000 nM T22717 CO32GA 25098140 IC50 = 410 nM T22717 CVF1L2 25098141 IC50 = 690 nM T22717 C75IZF 25098410 IC50 = 170 nM T22717 CT53KC 25098411 IC50 = 200 nM T22717 CY8WB9 25098412 IC50 = 290 nM T22717 CP03DL 57391543 IC50 = 60 nM T22717 CU48OP 57398520 IC50 > 5000 nM T22717 CB2DV7 57401984 IC50 > 5000 nM T22717 CL42OS 57402116 IC50 = 260 nM T22717 CBO25P 135412019 IC50 = 2570 nM T90070 D09BHB 5509 IC50 = 90 nM T90070 D0R1RS 3715 IC50 = 50 nM T90070 D0TG1H 3033 IC50 = 8 nM T90070 D0ZL4F 180540 IC50 = 20 nM T90070 CCZ3K9 15250 IC50 > 1000 nM T90070 C4PG1B 30931 IC50 > 1000 nM T90070 CNB6V7 114864 IC50 = 50 nM T90070 C7AKH8 141222 IC50 > 1000 nM T90070 C6EVL8 854057 IC50 > 1000 nM T90070 CNRE12 13309832 IC50 > 1000 nM T90070 CRB2H6 14762946 IC50 = 500 nM T90070 CNJ72V 18546323 IC50 > 1000 nM T90070 C5FD2Z 22218600 IC50 > 1000 nM T90070 CM3NT2 44298341 Ki = 13000 nM T90070 CX79VC 45268160 IC50 > 1000 nM T90070 C95IAE 45269044 IC50 = 600 nM T90070 CS2JM1 45269050 IC50 = 12 nM T90070 CEGP42 45269893 IC50 = 50 nM T90070 C5TE3O 45269894 IC50 = 13 nM T90070 C4O9EY 45269895 IC50 = 650 nM T90070 C34QNT 45269905 IC50 = 10 nM T90070 CGVT73 45270722 IC50 = 20 nM T90070 C4KH1C 45272452 IC50 = 25 nM T90070 C03KDJ 78224453 Ki = 7000 nM T90070 C0M8ZV 134130686 Ki = 106000 nM T90070 C1AS4F 134130687 Ki = 4000 nM T90070 CG0QB1 134130688 Ki = 12000 nM T90070 CFZG03 134130848 Ki = 10000 nM T90070 CGH9T1 134130849 Ki = 13000 nM T90070 CGW47R 134130850 Ki = 14000 nM T90070 C1NY6S 134130851 Ki = 6000 nM T90070 C2B3KN 134130852 Ki = 31000 nM T90070 CA0X3S 134130853 Ki = 4000 nM T90070 C42SCP 134130854 Ki = 383000 nM T90070 CD1TK0 134130855 Ki = 9300 nM T90070 CG35UE 134130856 Ki = 2300 nM T90070 D05EMX 14076674 IC50 = 25 nM T90070 D08GOT 13752584 IC50 = 400 nM T90070 D0I8YN 18546352 IC50 = 9 nM T90070 D0Q8ZV 15581854 IC50 = 500 nM T90070 D0T8RL 13409348 IC50 = 13 nM T39716 D00PEH 135449332 IC50 = 316227.77 nM T39716 D00STL 644241 IC50 = 1000000 nM T39716 D01AXB 60835 IC50 = 7943.28 nM T39716 D01AZG 5073 IC50 = 102000 nM T39716 D01FGR 3100 IC50 = 41000 nM T39716 D01UTL 2995 IC50 = 1520 nM T39716 D03DAP 3356 IC50 = 6500 nM T39716 D03FLC 3878 IC50 = 39810.72 nM T39716 D03HFG 5324346 IC50 = 39400 nM T39716 D03IGH 213039 IC50 = 39810.72 nM T39716 D03QWT 73303 IC50 = 1584893.19 nM T39716 D04FVU 6337614 IC50 = 19952.62 nM T39716 D04JEE 4946 IC50 = 2100 nM T39716 D05MQK 110635 IC50 = 125892.54 nM T39716 D05OFX 219078 IC50 = 501187.23 nM T39716 D08CDI 208908 IC50 = 3162277.66 nM T39716 D08HQK 5411 IC50 = 530 nM T39716 D09MWJ 2092 IC50 = 199526.23 nM T39716 D0B3UJ 115237 IC50 = 158489.32 nM T39716 D0BP9C 193962 IC50 = 501187.23 nM T39716 D0BZ7W 443879 IC50 = 6309.57 nM T39716 D0C7ET 11174599 IC50 > 30 nM T39716 D0C9SY 135400189 IC50 = 2511886.43 nM T39716 D0CL9S 159269 IC50 = 3162277.66 nM T39716 D0CS2F 3955 IC50 = 239 nM T39716 D0D7KC 5488548 IC50 = 251188.64 nM T39716 D0E4DW 1775 IC50 = 49000 nM T39716 D0E6XR 3062316 IC50 = 398107.17 nM T39716 D0H7KF 5002 IC50 = 16900 nM T39716 D0I1FQ 54671008 IC50 = 316227.77 nM T39716 D0J2KV 4932 IC50 = 1190 nM T39716 D0K3QS 6442177 IC50 = 199526.23 nM T39716 D0L4YD 154059 IC50 = 6309.57 nM T39716 D0NR6S 3002977 IC50 = 630957.34 nM T39716 D0NW3X 71329 IC50 > 300000 nM T39716 D0O3FG 125017 IC50 = 199526.23 nM T39716 D0Q5UQ 214348 IC50 = 79432.82 nM T39716 D0R0FE 2520 IC50 = 41500 nM T39716 D0R0MW 5329102 IC50 = 39810.72 nM T39716 D0U0VU 5312125 IC50 = 63095.73 nM T39716 D0U1OE 5452 IC50 = 1830 nM T39716 D0U2JP 4369359 IC50 = 630957.34 nM T39716 D0X0RI 4178 IC50 = 58000 nM T39716 D0X4RN 3676 IC50 = 108000 nM T39716 D0X5ZI 6918493 IC50 = 1000000 nM T39716 D0Y4JJ 2351 IC50 = 3700 nM T39716 D0Y5AM 444031 IC50 = 1584.89 nM T39716 D0Y5UG 2160 IC50 = 1600 nM T39716 D0Z1UA 71301 IC50 = 7943.28 nM T39716 D0Z7ZM 135398744 IC50 = 501187.23 nM T39716 D02AIN 122678117 IC50 > 33000 nM T39716 D04JZH 11659955 IC50 = 9000 nM T39716 D04PER 49836093 IC50 = 84 nM T39716 D06ENM 66553195 IC50 = 4700 nM T39716 D06TQR 76287260 IC50 > 100000 nM T39716 D0DH5X 44472635 IC50 > 30000 nM T39716 D0K9IF 71666749 IC50 > 30000 nM T39716 D0L9QM 59568713 IC50 > 30000 nM T39716 D0M3XR 46209133 IC50 > 30000 nM T39716 D0O7QA 46840946 IC50 = 11 nM T39716 D0OX9F 16046068 IC50 = 84000 nM T39716 D0P5CM 56945146 IC50 = 12589.25 nM T39716 D0S5IR 86294073 IC50 > 30000 nM T39716 D0W8XT 60663 IC50 = 500 nM T39716 D08IMD 16755780 IC50 = 14000 nM T39716 D0E2FZ 10149311 IC50 > 30000 nM T39716 D0HG2S 86294663 IC50 > 30000 nM T39716 D08SOF 5405 IC50 = 971 nM T39716 CZUI83 2769 IC50 = 14700 nM T39716 CP1QC0 9801 IC50 = 2520 nM T39716 C3H6AQ 21467 IC50 = 7800 nM T39716 CP8F7B 64143 IC50 = 501187.23 nM T39716 CLD6J9 441074 IC50 = 6900 nM T39716 CZN6S9 743974 IC50 > 100000 nM T39716 CPN25U 998021 IC50 = 9200 nM T39716 CTZ4R5 2730286 IC50 = 200 nM T39716 CORX94 2804997 IC50 = 5495.41 nM T39716 CMV0O1 3035569 IC50 = 30000 nM T39716 CM8IR4 4879545 IC50 = 980 nM T39716 C9ZT3K 9799052 IC50 = 2100 nM T39716 C5Z2KM 9805944 IC50 = 483 nM T39716 CY30OZ 9819588 IC50 = 2850 nM T39716 CS6FN7 9883254 IC50 = 8520 nM T39716 C4CH5D 9927877 IC50 = 4000 nM T39716 CREZ06 9928808 IC50 = 9000 nM T39716 CGY63T 10004877 IC50 > 100000 nM T39716 C5WLU0 10039502 IC50 = 5780 nM T39716 C1N5LX 10065677 IC50 = 13000 nM T39716 CF7OC8 10073954 IC50 = 30000 nM T39716 C97OQC 10088458 IC50 = 25000 nM T39716 C71ZGK 10316911 IC50 = 560 nM T39716 CT6Y9I 10365686 IC50 = 126000 nM T39716 C2KO8V 10388264 IC50 > 30000 nM T39716 CP7CH6 10389946 IC50 > 100000 nM T39716 CZN82G 10406083 IC50 = 15000 nM T39716 CBR9K8 11541314 IC50 = 60000 nM T39716 CS1V0J 11566989 IC50 = 2560 nM T39716 CKI9D5 11599973 IC50 > 31600 nM T39716 CQL5S8 11613750 IC50 > 100000 nM T39716 CXG1B4 11649741 IC50 > 100000 nM T39716 CH8K2V 11780892 IC50 > 100000 nM T39716 CD34SB 15982534 IC50 > 100000 nM T39716 CPCZ62 16040329 IC50 = 4700 nM T39716 CBF18D 21558498 IC50 = 455 nM T39716 CL73HJ 21589240 IC50 = 0.28 nM T39716 C5V2PF 22149197 IC50 = 14200 nM T39716 CAL57W 22149198 IC50 = 1510 nM T39716 CNM8X9 22149200 IC50 = 5250 nM T39716 C13HDG 22149207 IC50 = 5600 nM T39716 CYU64Q 22149216 IC50 = 8500 nM T39716 CUI6D7 22149230 IC50 = 8850 nM T39716 CNT32Z 22149267 IC50 = 2350 nM T39716 CH76LZ 22149271 IC50 = 1750 nM T39716 C2LUF7 22149278 IC50 = 7890 nM T39716 CL14RW 22149294 IC50 = 1100 nM T39716 CGBU69 22149297 IC50 = 4100 nM T39716 CMRN02 22149337 IC50 = 10800 nM T39716 CCY65J 22149344 IC50 = 3600 nM T39716 C6X0LN 22149356 IC50 = 3600 nM T39716 CFYW59 22149360 IC50 = 5400 nM T39716 CPXW92 22149373 IC50 = 2710 nM T39716 CUGR26 24757965 IC50 = 12000 nM T39716 CX79CS 24757966 IC50 > 30000 nM T39716 CDF15M 24759558 IC50 = 9000 nM T39716 CTG41H 24778289 IC50 > 2000 nM T39716 CM2DL3 24795066 IC50 > 30000 nM T39716 CF75YB 24857856 IC50 = 100 nM T39716 C3UNC4 24864147 IC50 = 14000 nM T39716 C6CK5U 24883321 IC50 = 4780 nM T39716 C5WOA3 24883322 IC50 = 7430 nM T39716 C5KA0N 24893979 IC50 = 84000 nM T39716 C21VCQ 25001553 IC50 = 7000 nM T39716 C6H4YL 25001554 IC50 = 25000 nM T39716 CUMH07 25001555 IC50 > 30000 nM T39716 CJR70I 25001557 IC50 = 26000 nM T39716 CIWR78 25001850 IC50 = 6000 nM T39716 C91QFN 25019282 IC50 > 30000 nM T39716 C0Z2SQ 25056787 IC50 = 2511.89 nM T39716 CPAZ91 25056788 IC50 = 5011.87 nM T39716 CP03LT 25113806 IC50 = 3981.07 nM T39716 CY5A6Q 25113809 IC50 = 3162.28 nM T39716 CK3JN1 25138309 IC50 = 7244.36 nM T39716 CWF5Z3 25143506 IC50 > 30000 nM T39716 CP72MB 25159060 IC50 = 12000 nM T39716 CBK27L 25196164 IC50 > 30000 nM T39716 CXKB13 25204469 IC50 = 8709.64 nM T39716 CAW05V 25204470 IC50 = 2630.27 nM T39716 C38CAX 25204471 IC50 > 25703.96 nM T39716 CUZ1Y2 25204472 IC50 = 8709.64 nM T39716 C1GO8L 25204473 IC50 = 1348.96 nM T39716 C9ZTJ3 25204533 IC50 > 15848.93 nM T39716 C2O6LT 25204534 IC50 > 33113.11 nM T39716 CBG48F 25204535 IC50 > 28840.32 nM T39716 C3JN6D 25204536 IC50 > 28183.83 nM T39716 C76UDL 25204600 IC50 = 8511.38 nM T39716 CXOZ41 25204603 IC50 = 5888.44 nM T39716 C08BDN 25204604 IC50 = 7762.47 nM T39716 C4IUB3 25204605 IC50 > 10471.29 nM T39716 CBH9O2 25204669 IC50 = 19952.62 nM T39716 C92WAR 25204670 IC50 > 33113.11 nM T39716 CYIV75 25204736 IC50 > 33113.11 nM T39716 CZY68S 25204738 IC50 > 33113.11 nM T39716 C1IW5M 25261456 IC50 > 10000 nM T39716 CY4LG8 42622934 IC50 > 30000 nM T39716 C96FIN 42644084 IC50 > 10000 nM T39716 C8BI5F 42644088 IC50 > 10000 nM T39716 CREJ31 42646199 IC50 > 10000 nM T39716 CKZ76R 42646202 IC50 < 10000 nM T39716 C81NVM 42646450 IC50 < 10000 nM T39716 CVBO78 42647178 IC50 < 10000 nM T39716 CX4YL8 44232522 IC50 > 10000 nM T39716 C7UY5F 44235863 IC50 > 10000 nM T39716 CX2W8Y 44236320 IC50 > 10000 nM T39716 C8LN0U 44236321 IC50 > 10000 nM T39716 CK4S5Y 44236322 IC50 > 10000 nM T39716 C62NRA 44337110 IC50 = 1760 nM T39716 C4K5MJ 44337198 IC50 = 15500 nM T39716 CP92BO 44337462 IC50 = 3920 nM T39716 CSMF57 44337512 IC50 = 10500 nM T39716 C85VGK 44337552 IC50 = 7900 nM T39716 C2QK4J 44472590 IC50 > 30000 nM T39716 CQ8C3F 44472591 IC50 > 30000 nM T39716 CC2TA5 44472592 IC50 > 30000 nM T39716 CWN95E 44472610 IC50 > 30000 nM T39716 C1H2ZT 44472612 IC50 > 30000 nM T39716 C9G5ID 44472613 IC50 > 30000 nM T39716 C5N4KE 44472633 IC50 > 30000 nM T39716 C5RNK0 44476261 IC50 = 4000 nM T39716 C6AK3W 44476911 IC50 > 30000 nM T39716 CLDQ43 44476913 IC50 > 30000 nM T39716 CG3R4T 44477000 IC50 = 27000 nM T39716 C1FTA7 44481065 IC50 > 30000 nM T39716 C01UWF 44540282 IC50 > 33000 nM T39716 CWP9Q3 44540283 IC50 > 33000 nM T39716 CKCG52 44540374 IC50 = 4400 nM T39716 CPFO82 44540469 IC50 = 18000 nM T39716 C46HBA 44540470 IC50 = 12000 nM T39716 C5NFE6 44540656 IC50 = 2900 nM T39716 C2MF7Z 44540754 IC50 = 4500 nM T39716 C5O4TM 44540839 IC50 = 19000 nM T39716 CYM71J 44543780 IC50 = 940 nM T39716 CD4LN9 44543781 IC50 = 2800 nM T39716 CE0K5T 44543783 IC50 = 12000 nM T39716 CS10AL 44543784 IC50 = 8700 nM T39716 C17LUC 44543889 IC50 = 4400 nM T39716 C9X2SL 44543890 IC50 > 26000 nM T39716 CE6HW8 44543891 IC50 = 6100 nM T39716 CB83EJ 44544123 IC50 > 31000 nM T39716 CN64WQ 44544347 IC50 = 730 nM T39716 CQ79RB 44544349 IC50 = 1600 nM T39716 CSV3F9 44544441 IC50 = 12000 nM T39716 C0RI5Z 44544444 IC50 = 3700 nM T39716 CK8T7U 44544546 IC50 = 8900 nM T39716 C7B0LF 44544548 IC50 = 8500 nM T39716 COJ7H6 44544644 IC50 = 6100 nM T39716 CYJB15 44544645 IC50 = 2600 nM T39716 CIO82A 44544649 IC50 > 23000 nM T39716 C8RAF0 44544851 IC50 = 19000 nM T39716 CWKZ36 44544853 IC50 > 8300 nM T39716 C6AX2C 44544950 IC50 = 4300 nM T39716 CGB50M 44545053 IC50 = 1900 nM T39716 C6VF4T 44545055 IC50 = 7900 nM T39716 CU16DA 44545166 IC50 = 16000 nM T39716 C9V7OF 44545167 IC50 > 33000 nM T39716 CW78UO 44545168 IC50 = 13000 nM T39716 CNZ12F 44545169 IC50 = 4700 nM T39716 CCD1V2 44545286 IC50 > 25000 nM T39716 C5KZ2M 44545289 IC50 = 1900 nM T39716 C9JK4V 44545402 IC50 = 17000 nM T39716 C6L8QO 44545403 IC50 = 810 nM T39716 CGLQ31 44552634 IC50 > 33000 nM T39716 CC2IO4 44552811 IC50 > 33000 nM T39716 CTX13C 44555196 IC50 > 33000 nM T39716 C5EX1K 44555473 IC50 > 10000 nM T39716 CXHT91 44571305 IC50 > 30000 nM T39716 CR32XZ 44571307 IC50 > 30000 nM T39716 C0IP7C 44583234 IC50 > 10000 nM T39716 C6HTC1 44583235 IC50 > 10000 nM T39716 CZJU04 44583236 IC50 < 10000 nM T39716 C3TYW0 44583237 IC50 < 10000 nM T39716 CCL9R0 44583238 IC50 > 10000 nM T39716 COX7F1 44583287 IC50 > 10000 nM T39716 C5SI9Q 44583288 IC50 > 10000 nM T39716 CFT74N 44583289 IC50 > 10000 nM T39716 CC19TZ 44583290 IC50 > 10000 nM T39716 C90RAV 44583349 IC50 > 10000 nM T39716 CK81NJ 44583350 IC50 > 10000 nM T39716 C20VTN 44583351 IC50 > 10000 nM T39716 CD5U3A 44583352 IC50 > 10000 nM T39716 C9G7VT 44583353 IC50 > 10000 nM T39716 C6QF4O 44583354 IC50 > 10000 nM T39716 C48AQR 44583355 IC50 > 10000 nM T39716 CG5X0M 44583356 IC50 < 10000 nM T39716 CUG9Y0 44583357 IC50 = 1000 nM T39716 CER76K 44585595 IC50 = 2300 nM T39716 C64ZKC 44593664 IC50 > 10000 nM T39716 C01BFQ 44593665 IC50 > 10000 nM T39716 C40BIM 45139151 IC50 = 15800 nM T39716 CUT2B4 45267348 IC50 > 10000 nM T39716 CJH3A2 45268206 IC50 > 10000 nM T39716 C4WR0V 45269087 IC50 > 10000 nM T39716 CRPS25 45269096 IC50 > 10000 nM T39716 C7BNY6 45269104 IC50 < 10000 nM T39716 CS1Q2X 45269947 IC50 > 10000 nM T39716 C1BE5U 45269948 IC50 > 10000 nM T39716 CG1H9N 45269950 IC50 = 10000 nM T39716 C1NT2M 45270771 IC50 > 10000 nM T39716 CA05IG 45270778 IC50 > 10000 nM T39716 CZ7MK9 45270788 IC50 < 10000 nM T39716 C9TM2P 45271593 IC50 > 10000 nM T39716 C06YAD 45271599 IC50 > 10000 nM T39716 CG0I8P 45271610 IC50 > 10000 nM T39716 C6FBH0 45271618 IC50 < 10000 nM T39716 C71VIG 45272510 IC50 > 10000 nM T39716 C05EDY 45272511 IC50 > 10000 nM T39716 CD62AH 45273373 IC50 > 10000 nM T39716 CMN39U 45273380 IC50 > 10000 nM T39716 C9L4KT 46205341 IC50 > 333000 nM T39716 CL41FE 46206000 IC50 > 333000 nM T39716 C1L0GS 46840949 IC50 = 17060 nM T39716 C4C0ED 46840950 IC50 > 10000 nM T39716 CI1YK3 46841216 IC50 = 35118 nM T39716 CD8M3F 46841499 IC50 = 29291 nM T39716 CO76ID 46841501 IC50 > 10000 nM T39716 CS5EJ1 46841648 IC50 > 30000 nM T39716 CRE97F 46841787 IC50 > 30000 nM T39716 COV0Q3 46841788 IC50 = 14413 nM T39716 C2OWF8 46841789 IC50 = 10549 nM T39716 CRU1P2 46882874 IC50 > 10000 nM T39716 C0FM2D 46882917 IC50 > 10000 nM T39716 CC1VO9 46882918 IC50 > 10000 nM T39716 C27RIV 46882919 IC50 > 10000 nM T39716 CE3O7D 46882949 IC50 > 10000 nM T39716 CHS1X0 46882950 IC50 > 10000 nM T39716 C3A1ZF 46882969 IC50 > 10000 nM T39716 CD7XA2 46882972 IC50 > 10000 nM T39716 CY5CW2 46882973 IC50 > 10000 nM T39716 C3ZPY7 46882986 IC50 > 10000 nM T39716 CKX8N2 46882987 IC50 > 10000 nM T39716 CG81CZ 46882988 IC50 > 10000 nM T39716 CP87CA 46883032 IC50 > 10000 nM T39716 CWU4T2 46883033 IC50 > 10000 nM T39716 C41RYD 46883034 IC50 > 10000 nM T39716 C3SQ2Z 46883035 IC50 > 10000 nM T39716 CS51UC 46883473 IC50 > 10000 nM T39716 CL0S4B 46883474 IC50 < 10000 nM T39716 C0K5ZJ 46883508 IC50 > 1000 nM T39716 CMNJ24 46883509 IC50 = 10000 nM T39716 CF4VC1 46883510 IC50 > 10000 nM T39716 C8Z0VS 49831248 IC50 = 351 nM T39716 C5LE0P 49850210 IC50 = 182 nM T39716 CLJ89W 49869305 IC50 = 1034 nM T39716 C9YM1Q 49869306 IC50 = 2938 nM T39716 CQ9PZ5 49869459 IC50 = 4577 nM T39716 C2N0XV 49869747 IC50 = 13770 nM T39716 C90UKY 50899643 IC50 > 30000 nM T39716 C94NCJ 50905973 IC50 = 223 nM T39716 CENW12 50925404 IC50 = 1320 nM T39716 C06OXV 52920492 IC50 = 69000 nM T39716 C6RFU2 53025800 IC50 = 4384 nM T39716 CPD0F2 53025889 IC50 = 7601 nM T39716 C0GF1R 53025891 IC50 = 4418 nM T39716 CMU7X8 53025901 IC50 = 7172 nM T39716 C08VWL 53025902 IC50 = 6943 nM T39716 CY74FO 53025906 IC50 = 8033 nM T39716 C5PB6K 53025909 IC50 = 4891 nM T39716 CY3R7J 53058099 IC50 = 4325 nM T39716 C8BG5J 53058100 IC50 = 3949 nM T39716 C02VSJ 53058119 IC50 = 8144 nM T39716 CK59VP 53058205 IC50 = 8092 nM T39716 CMS2F7 53239561 IC50 = 920 nM T39716 CRB6N5 53307604 IC50 > 33113.11 nM T39716 CJ83EB 53311393 IC50 > 10000 nM T39716 C23WVS 53361524 IC50 = 1100 nM T39716 C54YUZ 53362500 IC50 = 6800 nM T39716 CBAC86 53362558 IC50 = 500 nM T39716 CYX87Q 53362559 IC50 = 300 nM T39716 C8B1ZY 53362973 IC50 = 5400 nM T39716 CWA14L 53802926 IC50 > 6309.57 nM T39716 C28RDF 54746913 IC50 > 30000 nM T39716 CXEH21 56595883 IC50 = 1330 nM T39716 CSO3U5 56595888 IC50 = 541000 nM T39716 CY91VM 56595933 IC50 = 3300 nM T39716 CQ2J8B 56596030 IC50 = 2500 nM T39716 CY87LA 56596233 IC50 = 134000 nM T39716 CZ0K2U 56596475 IC50 = 215000 nM T39716 CXI5V1 56643481 IC50 > 5000 nM T39716 CH3BN6 56643486 IC50 > 5000 nM T39716 C6PUX9 56645570 IC50 > 30000 nM T39716 C6XI4W 56647652 IC50 > 5000 nM T39716 CG5T6R 56659661 IC50 > 33113.11 nM T39716 CUGJ21 56666584 IC50 > 33113.11 nM T39716 C39VWM 56676812 IC50 = 12022.64 nM T39716 C2LD6Y 56680137 IC50 = 4677.35 nM T39716 C5I4WJ 56680138 IC50 > 33113.11 nM T39716 CN5SE7 56683480 IC50 > 33113.11 nM T39716 C1IY0P 56944164 IC50 > 20000 nM T39716 CQT5I3 57328465 IC50 = 1260 nM T39716 CS1XE6 57328466 IC50 = 160 nM T39716 C4E1NK 57331209 IC50 > 30000 nM T39716 COUZ63 57494822 IC50 = 11102 nM T39716 C3N4MF 57520842 IC50 > 30000 nM T39716 CEL56T 57520942 IC50 > 30000 nM T39716 CR34CL 57582353 IC50 = 37000 nM T39716 C35GXV 57720515 EC50 = 29000 nM T39716 C09FAM 58044314 IC50 = 4000 nM T39716 CE3H1Q 58044315 IC50 > 10000 nM T39716 CZ28IJ 58044318 IC50 = 2500 nM T39716 CK0UY9 58044383 IC50 = 740000 nM T39716 CT4N2G 58044433 IC50 = 1903000 nM T39716 C2TRY9 58044589 IC50 = 1900 nM T39716 C0NFE7 58044606 IC50 = 981000 nM T39716 CF7PR9 58044619 IC50 = 3500 nM T39716 C9JCL7 58080768 IC50 = 10300 nM T39716 CRW9A3 58118918 IC50 = 102 nM T39716 C4FH0W 58118983 IC50 = 333 nM T39716 CCQM76 59153288 IC50 > 30000 nM T39716 CYF3R7 60167367 IC50 > 30000 nM T39716 C2D3HQ 60168069 IC50 > 100000 nM T39716 CSA3I9 60200914 IC50 = 1200 nM T39716 CK76WB 60200915 IC50 > 33000 nM T39716 CI40XK 60201083 IC50 = 19000 nM T39716 CNR41U 60201084 IC50 > 33000 nM T39716 CO5HD0 60201085 IC50 = 1200 nM T39716 CA57OQ 60201086 IC50 = 9700 nM T39716 C5UKQ8 60201087 IC50 = 25000 nM T39716 CA7NI3 60201088 IC50 > 16000 nM T39716 C56KOS 60201255 IC50 = 17000 nM T39716 C1YQ8J 60201256 IC50 > 25000 nM T39716 CVW28G 60201257 IC50 > 10000 nM T39716 CC82DM 65459349 IC50 = 27000 nM T39716 C6EJ3F 66551245 IC50 = 31622.78 nM T39716 C2LBW7 66551925 IC50 > 30000 nM T39716 CV7ZG3 66632452 IC50 = 3000 nM T39716 COTD35 66667669 IC50 = 11000 nM T39716 CD2HV3 66813354 IC50 > 31622.78 nM T39716 C78XLS 66813470 IC50 = 6309.57 nM T39716 CAOB97 66813557 IC50 = 3162.28 nM T39716 C89WUE 66813671 IC50 = 3981.07 nM T39716 CSY3F6 66813695 IC50 > 31622.78 nM T39716 CPK67V 66813703 IC50 > 31622.78 nM T39716 C7DX6Z 66813839 IC50 = 3981.07 nM T39716 CH2D5F 66813859 IC50 = 3162.28 nM T39716 C90OSR 66813870 IC50 = 7943.28 nM T39716 COZ0U9 66813914 IC50 = 6309.57 nM T39716 C5OTD2 66813927 IC50 = 5011.87 nM T39716 C39PEZ 66814019 IC50 = 3981.07 nM T39716 CG80RS 66814110 IC50 = 10000 nM T39716 C6QT5C 66849358 IC50 = 2221 nM T39716 CB2W9O 66849404 IC50 = 941 nM T39716 C7LOU6 66849415 IC50 = 8935 nM T39716 C4NZ5B 66849520 IC50 = 59 nM T39716 C6YC4U 66849571 IC50 = 887 nM T39716 CV9OX3 66849729 IC50 = 351 nM T39716 CWV2Z9 66849946 IC50 = 7541 nM T39716 CBQ5O1 67523614 IC50 = 1452 nM T39716 CM7AT3 67523656 IC50 = 1653 nM T39716 CB05ID 67972431 IC50 > 30000 nM T39716 CA7UZ6 68434755 IC50 > 30000 nM T39716 CBH6T3 69003776 IC50 = 14000 nM T39716 CXF5P9 69213151 IC50 = 1995.26 nM T39716 CP8XS4 70681040 IC50 = 360 nM T39716 CF85AB 70681063 IC50 = 120 nM T39716 C9LW7K 70681064 IC50 = 50 nM T39716 CX6UZ8 70681066 IC50 = 580 nM T39716 CS8V7G 70681068 IC50 = 150 nM T39716 CL28PN 70682458 IC50 = 10000 nM T39716 CJV64I 70683156 IC50 = 11800 nM T39716 C9BR3A 70683161 IC50 = 720 nM T39716 C36DYJ 70683164 IC50 = 2270 nM T39716 CN79ZX 70683165 IC50 = 780 nM T39716 CRXZ90 70683167 IC50 = 3000 nM T39716 C94GTH 70683168 IC50 = 460 nM T39716 C3ZY6F 70683178 IC50 = 50 nM T39716 C7NAV4 70683180 IC50 = 350 nM T39716 CN17AS 70683181 IC50 = 250 nM T39716 CA8VC6 70683182 IC50 = 130 nM T39716 C6QC5J 70683184 IC50 = 40 nM T39716 CK6JM8 70683187 IC50 = 60 nM T39716 CWK3H8 70683188 IC50 = 90 nM T39716 C1ARO8 70684544 IC50 = 6309.57 nM T39716 C3T1WM 70684545 IC50 > 31622.78 nM T39716 CIV4S6 70685239 IC50 = 1400 nM T39716 CLW68N 70685259 IC50 = 30 nM T39716 C65PTC 70685263 IC50 = 930 nM T39716 C2IDQ6 70685264 IC50 = 20 nM T39716 C02FWG 70685265 IC50 = 110 nM T39716 CO1ZR5 70685266 IC50 = 190 nM T39716 CRP7Z1 70685269 IC50 = 550 nM T39716 CRDJ83 70686683 IC50 = 19952.62 nM T39716 CEAK85 70687392 IC50 = 3700 nM T39716 CC32TO 70687393 IC50 = 1800 nM T39716 C0A3VH 70687418 IC50 = 40 nM T39716 CD2EW1 70688785 IC50 > 25118.86 nM T39716 C6YJL1 70689452 IC50 = 470 nM T39716 CO89VX 70689473 IC50 = 740 nM T39716 C56TAW 70689474 IC50 = 2700 nM T39716 CM3PD8 70689475 IC50 = 40 nM T39716 CV82BX 70690866 IC50 = 5011.87 nM T39716 C8R0SZ 70691558 IC50 = 590 nM T39716 CRXG05 70691559 IC50 = 1200 nM T39716 CYJ3F6 70691560 IC50 = 240 nM T39716 CK6I2V 70691577 IC50 = 80 nM T39716 C7ET5J 70691581 IC50 = 1570 nM T39716 CJ85NC 70691582 IC50 = 60 nM T39716 C27IPY 70691584 IC50 = 110 nM T39716 C8OKQ0 70693647 IC50 = 1700 nM T39716 CLN9F4 70693648 IC50 < 1000 nM T39716 CM3LU4 70693649 IC50 = 410 nM T39716 C3GVN0 70693667 IC50 = 200 nM T39716 CKP02Q 70693669 IC50 = 300 nM T39716 C6N3DT 70693670 IC50 = 2200 nM T39716 CEI84H 70693672 IC50 = 80 nM T39716 C6GCU1 70693673 IC50 = 30 nM T39716 CHUE45 70693674 IC50 = 80 nM T39716 CCQ49A 70695045 IC50 = 5011.87 nM T39716 CBCD89 70695046 IC50 = 5011.87 nM T39716 C63MTE 70695047 IC50 > 3162.28 nM T39716 CEK60M 70695761 IC50 = 500 nM T39716 CX6L3G 70695764 IC50 = 2000 nM T39716 CF4HZ3 70695774 IC50 = 120 nM T39716 CBHD70 70695780 IC50 = 140 nM T39716 CZL9G2 70695782 IC50 = 70 nM T39716 CKCE67 70695783 IC50 = 440 nM T39716 CUL37Y 70695784 IC50 = 90 nM T39716 C26OHM 70695785 IC50 = 20 nM T39716 CD1V2W 70695786 IC50 = 190 nM T39716 CBDL19 70792359 IC50 > 30000 nM T39716 CE9W1Z 70814180 IC50 = 6882 nM T39716 C7Z6HJ 70814238 IC50 = 8289 nM T39716 C7JD8A 70814244 IC50 = 9174 nM T39716 C1ST3M 70814308 IC50 = 4871 nM T39716 C5OT1G 70814333 IC50 = 9291 nM T39716 CLIH32 71226367 IC50 > 30000 nM T39716 C2FNI6 71259239 IC50 > 10000 nM T39716 CG0L7O 71259621 IC50 > 30000 nM T39716 C6BE5X 71271461 IC50 > 30000 nM T39716 CR4L9T 71449282 IC50 = 12589.25 nM T39716 CHF08N 71449283 IC50 = 6309.57 nM T39716 CMB7U1 71449284 IC50 = 6309.57 nM T39716 CVY54C 71449294 IC50 = 7943.28 nM T39716 C7L6QZ 71449295 IC50 > 31622.78 nM T39716 CIFE14 71451076 IC50 = 5011.87 nM T39716 CLSQ82 71451077 IC50 > 31622.78 nM T39716 C0RL3C 71451078 IC50 = 6309.57 nM T39716 CGJ7K0 71451084 IC50 = 19952.62 nM T39716 CI0B8V 71451085 IC50 = 1584.89 nM T39716 CXT57R 71452899 IC50 = 6309.57 nM T39716 CG21NF 71452900 IC50 > 31622.78 nM T39716 C7D9SN 71452907 IC50 > 31622.78 nM T39716 C5WU8L 71454670 IC50 = 5011.87 nM T39716 C7XQZ4 71454678 IC50 = 1000 nM T39716 CVU2O8 71454679 IC50 > 31622.78 nM T39716 C1X6TY 71456401 IC50 = 6309.57 nM T39716 C7AL1C 71456402 IC50 > 12589.25 nM T39716 CORH12 71456403 IC50 = 6309.57 nM T39716 C9FX5O 71456404 IC50 > 31622.78 nM T39716 CR4ZO3 71456412 IC50 = 794.33 nM T39716 CC3Q9J 71456413 IC50 = 2511.89 nM T39716 C7OW1B 71458245 IC50 > 31622.78 nM T39716 C6K4BO 71460096 IC50 > 31622.78 nM T39716 C9A7HP 71460097 IC50 > 31622.78 nM T39716 CYBR37 71460098 IC50 = 3162.28 nM T39716 CQW3L4 71460099 IC50 = 19952.62 nM T39716 CSB76D 71460108 IC50 = 1584.89 nM T39716 CQ30OU 71461829 IC50 > 31622.78 nM T39716 CV7ML5 71461830 IC50 = 10000 nM T39716 CA07TC 71517197 IC50 > 33000 nM T39716 CE60RK 71521279 IC50 = 4800 nM T39716 C5IK7D 71521280 IC50 = 5900 nM T39716 C2MC6B 71522734 IC50 > 10000 nM T39716 CM1B0W 71523649 IC50 = 36000 nM T39716 CHAU76 71555980 IC50 > 30000 nM T39716 C3EC1H 71557026 IC50 > 10000 nM T39716 CL85YK 71557177 IC50 > 10000 nM T39716 CY59CA 71557630 IC50 = 5200 nM T39716 CTI52S 71557789 IC50 > 10000 nM T39716 CO09GI 71558118 IC50 > 10000 nM T39716 CMKH30 71558122 IC50 > 10000 nM T39716 C48RIB 71558271 IC50 > 10000 nM T39716 CK2HF0 71558274 IC50 > 10000 nM T39716 CUI6M5 71558468 IC50 > 10000 nM T39716 C0DO9Y 71558578 IC50 > 10000 nM T39716 C2ZN4G 71558725 IC50 > 10000 nM T39716 CIDS01 71558883 IC50 > 10000 nM T39716 CY6Z1T 71558917 IC50 = 230 nM T39716 CHRO29 71558920 IC50 > 10000 nM T39716 C9WGA1 71559034 IC50 > 10000 nM T39716 C20ELR 71559363 IC50 > 10000 nM T39716 CJXK67 71559365 IC50 > 1000 nM T39716 CLAZ62 71585735 IC50 > 30000 nM T39716 CRC01X 71585929 IC50 = 5100 nM T39716 CXA29H 71585930 IC50 = 12000 nM T39716 CPI61F 71586033 IC50 > 30000 nM T39716 C4U3GM 71586128 IC50 > 30000 nM T39716 CNY52I 71586326 IC50 = 27000 nM T39716 C9J0EH 71603917 IC50 > 30000 nM T39716 C5LM0G 71711363 IC50 = 610 nM T39716 C1VC7P 71711696 IC50 = 4600 nM T39716 C8D7FJ 71711834 IC50 > 10000 nM T39716 CD4Z0Y 71711979 IC50 = 320 nM T39716 CK0L1B 71712241 IC50 > 10000 nM T39716 CZ5PL8 71716262 IC50 > 10000 nM T39716 C31BYG 71716276 IC50 > 30000 nM T39716 CC4A3K 71716821 IC50 = 43699 nM T39716 C7EG3T 71716825 IC50 = 25448 nM T39716 C9MUK3 71716856 IC50 = 15060 nM T39716 CUG2V3 71716866 IC50 > 30000 nM T39716 CIZ40M 71716873 IC50 > 10000 nM T39716 C4XYN9 71717494 IC50 = 22451 nM T39716 C0TK9Q 71718072 IC50 > 10000 nM T39716 C89GSF 71718127 IC50 > 30000 nM T39716 C7TM8H 71718630 IC50 > 10000 nM T39716 CW38FM 71718726 IC50 = 22210 nM T39716 CY6D2J 71719903 IC50 = 25786 nM T39716 CL0O5N 71719912 IC50 = 25231 nM T39716 CYQH30 71719914 IC50 > 30000 nM T39716 CMDI34 71720470 IC50 = 25578 nM T39716 C7B8UH 71720543 IC50 > 10000 nM T39716 C30NBJ 71722055 IC50 > 30000 nM T39716 C2QT3H 71812413 IC50 > 30000 nM T39716 CZPJ89 71812414 IC50 > 30000 nM T39716 CU1KS7 71812606 IC50 = 4000 nM T39716 CRAB14 71812607 IC50 = 11000 nM T39716 CQD1F2 71812796 IC50 = 24000 nM T39716 C2UOA5 71812797 IC50 = 28000 nM T39716 C9NK1C 71812798 IC50 > 30000 nM T39716 C3RE7M 71812799 IC50 > 30000 nM T39716 CW20HQ 71818431 IC50 = 50000 nM T39716 C2L7TX 71818575 IC50 = 3300 nM T39716 CYMS42 72545669 IC50 = 1070 nM T39716 C29YGC 72712370 IC50 = 9000 nM T39716 CCEX08 72949434 IC50 = 7200 nM T39716 C2E7QW 75201901 IC50 = 1100 nM T39716 C7OE1X 76309796 IC50 > 30000 nM T39716 CBH4N7 76309797 IC50 = 21000 nM T39716 C10UTF 76310404 IC50 > 30000 nM T39716 C6T1NV 76310406 IC50 > 30000 nM T39716 CC4BK5 76310408 IC50 = 20000 nM T39716 C8M7RN 76310409 IC50 > 30000 nM T39716 CHFC49 76313502 IC50 > 30000 nM T39716 C1PM7H 76314065 IC50 = 20000 nM T39716 CBK0T8 76314067 IC50 > 30000 nM T39716 C20ILA 76314069 IC50 > 30000 nM T39716 C8OQT1 76314070 IC50 = 27000 nM T39716 CNM4K0 76317019 IC50 > 30000 nM T39716 C32OSF 76317020 IC50 > 30000 nM T39716 CKG5A9 76317629 IC50 > 30000 nM T39716 CQ7JK4 76317631 IC50 > 30000 nM T39716 CT2R5J 76320732 IC50 > 30000 nM T39716 CVP8U9 76320733 IC50 > 30000 nM T39716 C2RJW0 76320734 IC50 > 30000 nM T39716 CY8NT4 76321352 IC50 > 30000 nM T39716 CRU30A 76321353 IC50 > 30000 nM T39716 CNY2D6 76321910 EC50 = 30000 nM T39716 CR05PL 76322043 IC50 > 30000 nM T39716 CQ3CW1 76322044 IC50 > 30000 nM T39716 C46MFT 76324385 IC50 > 30000 nM T39716 C4W1NV 76324386 IC50 = 20000 nM T39716 CJF20G 76324950 IC50 > 30000 nM T39716 CP3UI7 76327945 IC50 > 30000 nM T39716 CNY5X1 76328517 IC50 > 30000 nM T39716 CX54MA 76328518 IC50 > 30000 nM T39716 CINA95 76331591 IC50 > 30000 nM T39716 CCXK29 76332197 IC50 > 30000 nM T39716 CH4K7Q 76332198 IC50 > 30000 nM T39716 C4WO6Y 76332199 IC50 > 30000 nM T39716 CK47NO 76332200 IC50 > 30000 nM T39716 CANB89 76332201 IC50 > 30000 nM T39716 CO2N7R 76335221 IC50 > 30000 nM T39716 C05RSQ 76335223 IC50 > 30000 nM T39716 C8ND6L 76335224 IC50 = 21000 nM T39716 CUO84S 76335833 IC50 > 30000 nM T39716 C92WBQ 76336500 IC50 = 5600 nM T39716 C34TAM 77845572 IC50 > 30000 nM T39716 C2NCH9 78318214 IC50 > 30000 nM T39716 C2GET7 78318815 IC50 > 30000 nM T39716 C15BSO 86270136 IC50 = 265 nM T39716 CZL23E 86271138 IC50 > 30000 nM T39716 C7J9FE 86687346 IC50 = 21000 nM T39716 C0OTF5 86687356 IC50 = 21000 nM T39716 C50EDA 86687482 IC50 > 30000 nM T39716 CEQ0C1 86687530 IC50 > 30000 nM T39716 CTG76E 86687532 IC50 = 16000 nM T39716 CQN21C 86687557 IC50 > 30000 nM T39716 CFT89Y 86687602 IC50 = 1500 nM T39716 CY8JW3 86687604 IC50 > 10000 nM T39716 C7OXV8 86687606 IC50 > 10000 nM T39716 C63MCA 86687768 IC50 = 4750 nM T39716 CRJ9F2 86699098 IC50 > 10000 nM T39716 C4ZPG9 87178530 IC50 = 123 nM T39716 CHU2Z5 87178553 IC50 = 1647 nM T39716 CJ2OI4 87178572 IC50 = 211 nM T39716 CRHC58 87178657 IC50 = 281 nM T39716 CEH51J 87178674 IC50 = 166 nM T39716 C4FJ5M 87206909 IC50 = 397 nM T39716 CJC29A 89544489 IC50 > 10000 nM T39716 COK7U5 89545491 IC50 > 10000 nM T39716 CAM65C 89545507 IC50 > 10000 nM T39716 CMZ8P5 89545670 IC50 = 2600 nM T39716 C74SBC 89555961 IC50 > 10000 nM T39716 C01NKB 89555963 IC50 > 10000 nM T39716 C29LHS 89556026 IC50 > 10000 nM T39716 CXHC49 89556028 IC50 > 10000 nM T39716 CJRK20 89556063 IC50 > 10000 nM T39716 CH6AT7 89556066 IC50 = 5900 nM T39716 C9AMI1 89556077 IC50 > 10000 nM T39716 C72BSC 89556129 IC50 > 10000 nM T39716 CP8X3E 89573118 IC50 > 10000 nM T39716 C47HED 89583208 IC50 > 10000 nM T39716 CM6SL8 89613863 IC50 > 30000 nM T39716 CK8O4U 89614559 IC50 = 23000 nM T39716 C90UQK 89614650 IC50 > 30000 nM T39716 CQK1S9 89614770 IC50 > 30000 nM T39716 CV7UN4 89761281 IC50 = 1500 nM T39716 C7PT4Z 89761284 IC50 = 14000 nM T39716 CAO3I6 89761608 IC50 = 650 nM T39716 C29BFD 89761642 IC50 > 30000 nM T39716 CGI6O0 89761704 IC50 = 2100 nM T39716 C8IJ0Y 89761742 IC50 = 1500 nM T39716 C4BQC6 89761777 IC50 > 30000 nM T39716 COU52N 89761779 IC50 = 2000 nM T39716 C95IFK 89761981 IC50 > 30000 nM T39716 C48RCZ 90021555 IC50 = 1200 nM T39716 C1BIF8 90026208 IC50 = 50 nM T39716 C26LKW 90341025 IC50 > 30000 nM T39716 COYC71 90700276 IC50 = 1186 nM T39716 CN07GH 90846203 IC50 = 217 nM T39716 CX85KF 91134217 IC50 = 17810 nM T39716 C26BZK 91666633 IC50 = 110 nM T39716 C9ETC1 91666645 IC50 > 30000 nM T39716 C0S3JN 91799666 IC50 = 7200 nM T39716 C7NLE8 91809347 IC50 = 49 nM T39716 CTS64R 91809389 IC50 = 22000 nM T39716 CXN69G 100657083 IC50 = 1300 nM T39716 CQ9PN8 102593934 IC50 > 100000 nM T39716 CNFW42 117608566 IC50 = 1313 nM T39716 CC5N9I 117737142 IC50 > 14000 nM T39716 C4NH6M 117740584 IC50 > 10000 nM T39716 CC1A0T 117741702 IC50 > 10000 nM T39716 C3C2YG 117741784 IC50 > 10000 nM T39716 C4ZO0A 117741876 IC50 > 10000 nM T39716 C10BKY 117749324 IC50 > 30000 nM T39716 COVX65 117753917 IC50 > 10000 nM T39716 CS5X4R 117753922 IC50 = 140 nM T39716 CQK1U5 117753939 IC50 = 820 nM T39716 CW8RS3 117760464 IC50 > 30000 nM T39716 C3P1LN 117789501 IC50 = 419 nM T39716 CK0RV9 117993874 IC50 = 18000 nM T39716 CL4O0J 117993881 IC50 = 18800 nM T39716 CB8I3S 117993884 IC50 = 11000 nM T39716 C92RVJ 117993886 IC50 = 6000 nM T39716 CM2H5Q 117993976 IC50 = 2350 nM T39716 C9KV7L 117993993 IC50 = 6900 nM T39716 CNV24M 117993998 IC50 > 30000 nM T39716 C8DSV0 117994021 IC50 = 21000 nM T39716 C57PMF 118002063 IC50 = 32000 nM T39716 CT8C0X 118109014 IC50 = 5700 nM T39716 COH9J3 118109161 IC50 > 30000 nM T39716 CG3M4J 118109168 IC50 = 19000 nM T39716 CO6KX7 118109201 IC50 > 30000 nM T39716 CAU5T9 118109234 IC50 > 30000 nM T39716 CT4ZN7 118109256 IC50 > 30000 nM T39716 CG8FJ5 118109302 IC50 > 30000 nM T39716 C8OAL5 118109304 IC50 > 30000 nM T39716 C3N0KS 118109319 IC50 = 24200 nM T39716 CU85FO 118109356 IC50 = 1900 nM T39716 CWJ7T6 118109371 IC50 = 17600 nM T39716 CS0B7V 118112295 IC50 > 30000 nM T39716 CWR6I1 118112300 IC50 = 2.2 nM T39716 CXY23I 118121135 IC50 > 30000 nM T39716 CB4I7H 118121139 IC50 = 22500 nM T39716 C7AYV5 118540795 IC50 = 2000 nM T39716 CKA2F8 118554582 IC50 > 3000 nM T39716 C2O7GE 118707553 IC50 > 33000 nM T39716 C8S9VW 118707562 IC50 > 33000 nM T39716 CR8TX9 118708662 IC50 = 79 nM T39716 CMDN36 118710321 IC50 = 9716 nM T39716 CPL32R 118710322 IC50 = 12875 nM T39716 CA79ZM 118710323 IC50 > 30000 nM T39716 CLS68B 118710324 IC50 = 947 nM T39716 CL2PK9 118710325 IC50 = 7240 nM T39716 CDO95Z 118710326 IC50 = 572 nM T39716 CG7X9J 118710327 IC50 = 934 nM T39716 C83LIE 118710328 IC50 = 1329 nM T39716 CH29DT 118711022 IC50 = 24700 nM T39716 C3BQM2 118714771 IC50 = 181 nM T39716 CPVC71 118714772 IC50 = 340 nM T39716 CEB6T7 118714773 IC50 = 2216 nM T39716 C65NKL 118714774 IC50 = 358 nM T39716 C39NSR 118714775 IC50 = 3261 nM T39716 CJ8E7U 118714776 IC50 = 519 nM T39716 C84KNW 118714777 IC50 = 30000 nM T39716 CHS5K3 118714778 IC50 = 3069 nM T39716 C58YHZ 118714779 IC50 = 2450 nM T39716 CF2YQ4 118714780 IC50 = 30000 nM T39716 C40SOZ 118714781 IC50 = 1138 nM T39716 C67FSV 118714782 IC50 = 118 nM T39716 CREM47 118714783 IC50 = 1732 nM T39716 CX4I5Q 118714784 IC50 = 2811 nM T39716 CC56DO 118718808 IC50 > 30000 nM T39716 C69PLO 118734433 IC50 > 5000 nM T39716 C2NAE8 118734434 IC50 > 5000 nM T39716 CD4B5E 118734435 IC50 > 5000 nM T39716 C91PCO 118734436 IC50 > 5000 nM T39716 CM2Y6W 118734437 IC50 = 27000 nM T39716 CFL60J 118734438 IC50 > 5000 nM T39716 CQ0R3E 118734439 IC50 > 5000 nM T39716 CY8A1T 118734440 IC50 > 5000 nM T39716 CFRZ45 118734441 IC50 > 5000 nM T39716 C3ZJ0K 118734442 IC50 > 5000 nM T39716 CI30YK 118734443 IC50 > 5000 nM T39716 CUAQ60 118734444 IC50 > 5000 nM T39716 CFNR84 118734445 IC50 > 5000 nM T39716 CK12TX 118734446 IC50 > 20000 nM T39716 C09BDT 118734447 IC50 > 20000 nM T39716 C6F9BI 118734448 IC50 > 5000 nM T39716 C8ZLX9 118734449 IC50 > 20000 nM T39716 C01BNE 118734450 IC50 > 5000 nM T39716 CI0FE2 118734451 IC50 > 4700 nM T39716 C1CED0 118734452 IC50 > 5000 nM T39716 C8NBL5 118734453 IC50 > 5000 nM T39716 C0CY2K 118734454 IC50 > 5000 nM T39716 CTR7O8 118734455 IC50 > 5000 nM T39716 CZQD84 118734456 IC50 > 5000 nM T39716 CGBF25 118734457 IC50 > 5000 nM T39716 C6I8HF 118734458 IC50 > 5000 nM T39716 C5G7DQ 118734459 IC50 > 5000 nM T39716 CVW15D 118734460 IC50 > 5000 nM T39716 CSE60C 118734461 IC50 > 5000 nM T39716 CO4U1R 118734462 IC50 > 10000 nM T39716 CA95IF 118734463 IC50 > 10000 nM T39716 C14ILF 118734464 IC50 > 10000 nM T39716 C3TOV9 118734465 IC50 > 10000 nM T39716 C2RO8T 118734466 IC50 > 10000 nM T39716 CSP25D 118734467 IC50 > 10000 nM T39716 CJD80C 118734468 IC50 > 10000 nM T39716 C06TAI 118734469 IC50 > 10000 nM T39716 CBY5M0 118734470 IC50 > 10000 nM T39716 CHO8I3 118734471 IC50 = 3500 nM T39716 C38BCH 118734472 IC50 > 10000 nM T39716 CV7UH5 118734473 IC50 > 10000 nM T39716 C6SEA7 118734474 IC50 > 10000 nM T39716 CO7DP2 118734475 IC50 = 2100 nM T39716 CX2R0E 118734476 IC50 = 1100 nM T39716 C16AEK 118734477 IC50 > 10000 nM T39716 CO1UF9 118734478 IC50 = 2800 nM T39716 C16AUM 118734479 IC50 = 3000 nM T39716 CI2P1V 118734480 IC50 > 10000 nM T39716 C1Z8AN 118734481 IC50 = 3400 nM T39716 CYD8N6 118734482 IC50 = 400 nM T39716 CW05LY 118734483 IC50 > 10000 nM T39716 CN01US 118734484 IC50 > 10000 nM T39716 C3E7GP 118734485 IC50 > 10000 nM T39716 CCA41Z 118734486 IC50 > 10000 nM T39716 CM2QS5 118734487 IC50 = 3600 nM T39716 C3T1QC 118734488 IC50 = 4600 nM T39716 CM6Y8X 118734489 IC50 = 500 nM T39716 C93LMC 118734490 IC50 > 10000 nM T39716 C8LHA3 118734491 IC50 = 4500 nM T39716 C26ADB 118734547 IC50 = 8800 nM T39716 C82UBF 118734548 IC50 > 10000 nM T39716 CO4KD2 118734549 IC50 > 10000 nM T39716 CX6L4C 118734550 IC50 > 10000 nM T39716 C5JNX2 118734551 IC50 > 10000 nM T39716 C0UJ8Q 118734552 IC50 > 10000 nM T39716 CJDP52 118734553 IC50 > 10000 nM T39716 CM59EQ 118917669 IC50 > 100000 nM T39716 C6J8YF 118917671 IC50 > 30000 nM T39716 C0RFQ5 118937646 IC50 = 14200 nM T39716 CTR37C 118937656 IC50 > 33000 nM T39716 CTC20B 118937664 IC50 = 19000 nM T39716 CR9Y6M 118937702 IC50 = 3100 nM T39716 C1Y7MU 118937716 IC50 = 23000 nM T39716 C9JL4Y 118937760 IC50 > 33000 nM T39716 CXI1F9 118937849 IC50 > 33000 nM T39716 CWL1S3 118937903 IC50 > 33000 nM T39716 CXZ43S 118937913 IC50 = 5000 nM T39716 CMQB61 118937925 IC50 = 15000 nM T39716 CU4CW1 121313969 IC50 > 30000 nM T39716 C9H0BR 121333853 IC50 > 10000 nM T39716 CGH4B7 121333855 IC50 > 10000 nM T39716 CZ3X9J 121333858 IC50 > 10000 nM T39716 CT4FA9 121333871 IC50 > 10000 nM T39716 CIQ8C0 121333899 IC50 > 10000 nM T39716 C83STC 121333902 IC50 > 10000 nM T39716 CMA2O3 121333930 IC50 > 10000 nM T39716 C9Q2ND 121333973 IC50 = 12000 nM T39716 CO9SQ6 121454909 IC50 > 30000 nM T39716 CH0X4Z 121454982 IC50 > 30000 nM T39716 CT0KS4 121455652 IC50 > 30000 nM T39716 CW35TI 121455794 IC50 > 30000 nM T39716 CHD26A 121596332 IC50 > 33300 nM T39716 CNGQ19 122179477 IC50 > 30000 nM T39716 C1XKA8 122191834 IC50 > 30000 nM T39716 CHPL50 122194669 IC50 = 4400 nM T39716 CWSA14 122194670 IC50 = 2800 nM T39716 C05AUF 122194671 IC50 = 5600 nM T39716 CY2B6W 122194672 IC50 = 3000 nM T39716 CP38IW 122194673 IC50 = 6100 nM T39716 CWGY65 122194675 IC50 = 1100 nM T39716 C1MH8Y 122194676 IC50 = 3400 nM T39716 CP4L5A 122194677 IC50 = 16000 nM T39716 CW3D9H 122196008 IC50 = 20000 nM T39716 C5G9FH 122196009 IC50 = 7000 nM T39716 C2RBF4 122196010 IC50 = 17000 nM T39716 C0R8OS 122196011 IC50 = 18000 nM T39716 C61QNK 122196012 IC50 > 33000 nM T39716 CZ2HR6 122196013 IC50 = 5200 nM T39716 C6W5IA 122196014 IC50 = 3400 nM T39716 CKEH54 122196015 IC50 = 33000 nM T39716 C38XFL 122196016 IC50 = 24000 nM T39716 CLQ8O5 122196017 IC50 = 4900 nM T39716 C82UNL 122196018 IC50 = 1900 nM T39716 C0KG7Z 122196019 IC50 = 3700 nM T39716 CS0W4O 122196020 IC50 = 1200 nM T39716 CK8FH3 122196021 IC50 = 38000 nM T39716 C9N1CF 122196022 IC50 = 77000 nM T39716 CR4JT9 122196023 IC50 = 10000 nM T39716 C80OZQ 122196024 IC50 = 13000 nM T39716 CT9N7O 122196025 IC50 = 7100 nM T39716 C3B0RY 122422350 IC50 = 2500 nM T39716 C81EPB 122422402 IC50 = 23700 nM T39716 CC2TE4 122422536 IC50 = 16100 nM T39716 CEGS87 122513481 IC50 = 16400 nM T39716 C9K5RV 122513516 IC50 > 33000 nM T39716 CC1J0T 122591381 IC50 > 30000 nM T39716 C1YK2E 122678192 IC50 > 33000 nM T39716 C4D9QY 127026491 IC50 > 30000 nM T39716 C7L1DB 127037832 IC50 > 30000 nM T39716 CB98DL 127044262 IC50 = 7915 nM T39716 CZF2X5 127044562 IC50 = 5052 nM T39716 C4WEA5 127044563 IC50 = 425 nM T39716 C5J3AM 127044564 IC50 = 417 nM T39716 CE7MG6 127044736 IC50 > 10000 nM T39716 CMF6K2 127044897 IC50 = 353 nM T39716 CJC30T 127044898 IC50 = 3345 nM T39716 CXEZ15 127044899 IC50 = 1512 nM T39716 CYVO30 127045496 IC50 = 901 nM T39716 C7JT8V 127045799 IC50 > 5000 nM T39716 CH2Z3S 127045806 IC50 > 5000 nM T39716 CSJD60 127045808 IC50 > 4800 nM T39716 COWD91 127045811 IC50 > 10000 nM T39716 C90JPN 127045813 IC50 > 5000 nM T39716 C21JCE 127045825 IC50 > 5000 nM T39716 CNF0G1 127045829 IC50 > 5000 nM T39716 CC9TY3 127045830 IC50 > 5000 nM T39716 CDC0M9 127046018 IC50 > 5000 nM T39716 C74SHI 127046022 IC50 > 5000 nM T39716 CH0CD1 127046023 IC50 > 5000 nM T39716 CPX1F0 127046025 IC50 > 5000 nM T39716 CAVD37 127046026 IC50 > 5000 nM T39716 C8UW6X 127046032 IC50 = 900 nM T39716 CMPZ51 127046033 IC50 > 5000 nM T39716 CY5J0R 127046039 IC50 > 5000 nM T39716 CBQ47D 127046045 IC50 > 5000 nM T39716 C6NVQ1 127046047 IC50 > 5000 nM T39716 C4MU2J 127046230 IC50 > 5000 nM T39716 CGYE23 127046231 IC50 > 5000 nM T39716 C69GBJ 127046239 IC50 > 5000 nM T39716 CM1IH3 127046241 IC50 > 5000 nM T39716 C4L1VA 127046242 IC50 > 5000 nM T39716 CWN2J7 127046243 IC50 > 5000 nM T39716 CI1VA2 127046252 IC50 = 15900 nM T39716 CE67AD 127046253 IC50 = 1000 nM T39716 C53RIX 127046257 IC50 > 5000 nM T39716 COK9Z3 127046259 IC50 > 5000 nM T39716 CL5VY9 127046359 IC50 = 1800 nM T39716 C3M6YT 127046415 IC50 > 5000 nM T39716 C90HYR 127046420 IC50 > 5000 nM T39716 C8BES0 127046422 IC50 > 10000 nM T39716 C2EI4Q 127046423 IC50 = 37900 nM T39716 CM2HB0 127046424 IC50 > 5000 nM T39716 CM5D6J 127046425 IC50 > 5000 nM T39716 C9LH4U 127046428 IC50 > 5000 nM T39716 C20KGH 127046429 IC50 > 5000 nM T39716 CH27MP 127046433 IC50 > 5000 nM T39716 CWH7Y0 127046434 IC50 > 5000 nM T39716 C1CV8E 127046436 IC50 > 5000 nM T39716 C87YLU 127046583 IC50 > 5000 nM T39716 C74ELB 127046587 IC50 > 5000 nM T39716 CI9XY7 127046589 IC50 > 5000 nM T39716 CQ3EV4 127046592 IC50 > 5000 nM T39716 C8PO4C 127046597 IC50 = 22700 nM T39716 C31XHN 127046598 IC50 > 5000 nM T39716 CFSH84 127046606 IC50 > 5000 nM T39716 CP8T2D 127046764 IC50 > 5000 nM T39716 C0A7SK 127046767 IC50 > 5000 nM T39716 CC2Y1J 127046770 IC50 > 5000 nM T39716 C1XON9 127046774 IC50 > 5000 nM T39716 C80RLU 127046781 IC50 > 5000 nM T39716 C34GAN 127046799 IC50 = 2000 nM T39716 CCXR80 127046802 IC50 = 3400 nM T39716 CSKX63 127046908 IC50 > 5000 nM T39716 CVUW94 127046909 IC50 = 3200 nM T39716 C02HPV 127046912 IC50 > 2700 nM T39716 C8CK6P 127046914 IC50 > 5000 nM T39716 C3CSI0 127046916 IC50 = 4500 nM T39716 C4X2OU 127046919 IC50 > 5000 nM T39716 CL9W8T 127046920 IC50 > 5000 nM T39716 CLH51Y 127046923 IC50 > 5000 nM T39716 CXMC23 127046930 IC50 > 5000 nM T39716 CB9EF5 127046932 IC50 > 4800 nM T39716 CZ7G6T 127047057 IC50 > 5000 nM T39716 CND20E 127047062 IC50 > 5000 nM T39716 CNSZ83 127047063 IC50 > 5000 nM T39716 C1R4VN 127047068 IC50 > 5000 nM T39716 C5VU7H 127047069 IC50 > 5000 nM T39716 CFG94A 127047073 IC50 > 5000 nM T39716 CF5D0S 127047074 IC50 > 5000 nM T39716 C0XS7B 127047075 IC50 > 5000 nM T39716 CI60KD 127047206 IC50 > 10000 nM T39716 CA7YG4 127047208 IC50 > 5000 nM T39716 CXT5Y0 127047216 IC50 > 5000 nM T39716 CY8RH9 127047220 IC50 > 5000 nM T39716 CV4OB1 127047223 IC50 > 5000 nM T39716 C1RD6X 127047251 IC50 = 4400 nM T39716 CZLT12 127047252 IC50 = 2500 nM T39716 CFPJ73 127047320 IC50 > 5000 nM T39716 C3JK6P 127047322 IC50 > 5000 nM T39716 C1T5PC 127047323 IC50 > 5000 nM T39716 C28REX 127047327 IC50 > 5000 nM T39716 CVSF19 127047330 IC50 > 5000 nM T39716 C0IO2K 127047331 IC50 > 5000 nM T39716 C9SIK3 127047333 IC50 > 5000 nM T39716 CKD78E 127047346 IC50 = 3600 nM T39716 C5DO7I 127047347 IC50 > 5000 nM T39716 CM5TX2 127047468 IC50 > 5000 nM T39716 C54TRJ 127047469 IC50 > 5000 nM T39716 C3K5YI 127047471 IC50 > 5000 nM T39716 C2M5JH 127047472 IC50 > 5000 nM T39716 C3SLJ4 127047473 IC50 > 5000 nM T39716 CCA51M 127047474 IC50 = 7800 nM T39716 C6EM0G 127047476 IC50 > 5000 nM T39716 C5RKB7 127047479 IC50 > 4700 nM T39716 C96VDX 127047480 IC50 > 5000 nM T39716 CJ7IQ4 127047485 IC50 > 4000 nM T39716 CZKB91 127047487 IC50 > 5000 nM T39716 C7OTX3 127047488 IC50 > 5000 nM T39716 CVR95B 127047489 IC50 > 5000 nM T39716 CW8P5Y 127047613 IC50 > 5000 nM T39716 C0WXP3 127047615 IC50 > 5000 nM T39716 C1RK5C 127047619 IC50 > 5000 nM T39716 C9QZH7 127047622 IC50 > 5000 nM T39716 CJ31BC 127047628 IC50 > 5000 nM T39716 C9MXK5 127047633 IC50 > 5000 nM T39716 CB16MW 127047643 IC50 = 1000 nM T39716 C09QIY 127047645 IC50 = 2800 nM T39716 C5S1AI 127047646 IC50 = 5100 nM T39716 C1ULZ3 127047735 IC50 > 5000 nM T39716 C4T5WS 127047736 IC50 > 5000 nM T39716 CQ45AO 127047757 IC50 > 5000 nM T39716 CG5X0Y 127047758 IC50 = 5000 nM T39716 CTRE63 127047854 IC50 > 5000 nM T39716 CDGS14 127047866 IC50 > 5000 nM T39716 C16NUB 127047867 IC50 > 5000 nM T39716 CG52RP 127047873 IC50 > 5000 nM T39716 C8PWL6 127047983 IC50 > 5000 nM T39716 CGW63M 127047988 IC50 > 5000 nM T39716 CR6AB0 127047989 IC50 > 5000 nM T39716 CK9ZO8 127047990 IC50 > 5000 nM T39716 CQ2SO8 127047999 IC50 > 10000 nM T39716 C2D9LN 127048108 IC50 > 10000 nM T39716 C25GJD 127048113 IC50 = 3400 nM T39716 C4VID9 127048115 IC50 > 5000 nM T39716 CCI81A 127048120 IC50 > 5000 nM T39716 CE1Z4W 127048121 IC50 = 3400 nM T39716 CI0P1M 127048127 IC50 > 5000 nM T39716 C4CUP9 127048128 IC50 > 5000 nM T39716 C7HGD0 127048130 IC50 > 5000 nM T39716 C4LK6A 127048137 IC50 > 5000 nM T39716 CNA30T 127048138 IC50 > 5000 nM T39716 C38WDU 129012089 IC50 = 13000 nM T39716 C4Z5MQ 131839619 IC50 > 30000 nM T39716 C4A2JF 132020399 IC50 = 15105 nM T39716 C9C5PT 132020406 IC50 > 30000 nM T39716 COH0K2 132020407 IC50 = 18000 nM T39716 CX6WL3 132020408 IC50 > 30000 nM T39716 CABH81 132020419 IC50 > 30000 nM T39716 C79BLN 132020421 IC50 = 6300 nM T39716 CZ5H2B 132020452 IC50 = 18347 nM T39716 CNK15D 132020464 IC50 = 16000 nM T39716 CMD5X6 132020466 IC50 = 14000 nM T39716 C4FPR1 132020468 IC50 > 30000 nM T39716 CTRG94 132020475 IC50 > 30000 nM T39716 C76RHU 132020480 IC50 = 8600 nM T39716 C6ME9R 132020486 IC50 = 24000 nM T39716 C69ELN 132020488 IC50 = 1700 nM T39716 CIM31O 132020491 IC50 = 5700 nM T39716 CB74IC 132020507 IC50 = 12000 nM T39716 C4JP3T 132020512 IC50 > 30000 nM T39716 CDL95F 132020518 IC50 = 20000 nM T39716 CUZ03K 132020526 IC50 = 9666 nM T39716 CD4HS0 132020533 IC50 = 3900 nM T39716 C5LYQ6 132020541 IC50 = 30000 nM T39716 C5G1PQ 132020544 IC50 = 8400 nM T39716 CAZI64 132020570 IC50 = 3697 nM T39716 CTC7E3 132020571 IC50 = 6508 nM T39716 CP8A1Q 132020575 IC50 = 16000 nM T39716 C7ZIP5 132020580 IC50 = 7500 nM T39716 CLV79P 132020582 IC50 = 5100 nM T39716 CF2QM1 132020584 IC50 = 7200 nM T39716 CM42HK 132020589 IC50 > 30000 nM T39716 C21QHW 132051336 IC50 = 18000 nM T39716 C9RBP0 132051461 IC50 > 30000 nM T39716 CVFK13 132051462 IC50 > 30000 nM T39716 CNZA27 132051626 IC50 > 30000 nM T39716 CHL97M 132051650 IC50 = 11000 nM T39716 C83UBM 132051677 IC50 = 3800 nM T39716 CG1S2M 132519335 IC50 = 13000 nM T39716 CO2SH1 132519336 IC50 = 13000 nM T39716 CO1RW6 134132142 IC50 = 9134 nM T39716 CF2M4S 134132899 IC50 = 21000 nM T39716 C1M8ZR 134133921 IC50 > 30000 nM T39716 CJOQ95 134134229 IC50 > 30000 nM T39716 CC7OQ2 134135307 IC50 > 30000 nM T39716 CE5TV4 134135453 IC50 = 21000 nM T39716 CN7RI4 134146511 IC50 > 30000 nM T39716 CA5B2J 134150245 IC50 = 17430 nM T39716 COPA84 134151189 IC50 > 30000 nM T39716 CA49BH 134156727 IC50 = 27000 nM T39716 CFR87X 134477051 IC50 = 74 nM T39716 CFYC29 134477061 IC50 > 30000 nM T39716 C20QBE 134477062 IC50 = 1900 nM T39716 CT58HM 134477070 IC50 > 30000 nM T39716 C8W9YN 134477076 IC50 = 108 nM T39716 CX5MS3 134477080 IC50 = 50 nM T39716 CSO3Q9 134477081 IC50 = 37 nM T39716 CAED75 134477093 IC50 > 30000 nM T39716 CO15IT 134477094 IC50 > 30000 nM T39716 C0Q1MD 134477108 IC50 > 30000 nM T39716 CX64SG 134477133 IC50 > 30000 nM T39716 CT7J4U 134477136 IC50 > 30000 nM T39716 C51SKX 134477137 IC50 = 120 nM T39716 CCVX65 134477139 IC50 = 156 nM T39716 C03SFG 134477143 IC50 > 30000 nM T39716 C70XMC 134477147 IC50 > 30000 nM T39716 C7JM1E 134477177 IC50 = 5100 nM T39716 C4LS2A 134477178 IC50 = 2600 nM T39716 CNU8M6 134477183 IC50 = 133 nM T39716 CK9SR3 134477213 IC50 = 127 nM T39716 C9WN3E 134477214 IC50 = 4900 nM T39716 C9IB8P 134477217 IC50 > 30000 nM T39716 C1AB5Q 134477222 IC50 = 189 nM T39716 CN37XZ 134477224 IC50 > 30000 nM T39716 CR39TS 134477260 IC50 > 30000 nM T39716 C9O5FS 134477264 IC50 = 237 nM T39716 CS5ME8 134477268 IC50 = 150 nM T39716 CC0OF9 134477275 IC50 = 188 nM T39716 C1R9DV 134477283 IC50 > 30000 nM T39716 CMH4G1 135412290 IC50 = 1200 nM T39716 CB1VD9 135426471 IC50 = 300 nM T39716 CZ6WT3 135469086 IC50 = 19700 nM T39716 CY4MV6 135566354 IC50 > 30000 nM T39716 CMC7Q6 135568488 IC50 = 4500 nM T39716 C3YB0A 135568523 IC50 = 24350 nM T39716 CL43OY 135568535 IC50 = 5750 nM T39716 C4OVP2 136416802 IC50 > 30000 nM T39716 C7ZCT8 136416815 IC50 > 30000 nM T39716 C6B5US 137628648 IC50 > 10000 nM T39716 C2QCA5 137631487 IC50 > 30000 nM T39716 C8JA9G 137631733 IC50 > 30000 nM T39716 CB4A0Y 137632255 IC50 = 3200 nM T39716 C2XI8Y 137632393 IC50 > 30000 nM T39716 CES7L0 137632608 IC50 = 874 nM T39716 C28PMQ 137634084 IC50 = 6500 nM T39716 C8HPN4 137634334 IC50 > 30000 nM T39716 CLG25H 137634494 IC50 > 30000 nM T39716 C7S8YV 137636062 IC50 = 444 nM T39716 C08DOT 137636231 IC50 = 480 nM T39716 CM51CG 137636524 IC50 = 156 nM T39716 CNA56O 137636856 IC50 = 336 nM T39716 CO3QJ8 137637393 IC50 = 1200 nM T39716 CJH2V9 137637559 IC50 = 18200 nM T39716 CH3M0S 137637752 IC50 = 260 nM T39716 CFK9D8 137638117 IC50 = 169 nM T39716 C8EZ4N 137638256 IC50 = 6400 nM T39716 CW95QX 137638418 IC50 = 3900 nM T39716 CEP37F 137638536 IC50 > 30000 nM T39716 CLEF51 137638686 IC50 = 12800 nM T39716 C0ZS9N 137638993 IC50 = 76 nM T39716 C5KEW7 137639838 IC50 = 931 nM T39716 CK1C5F 137640087 IC50 > 10000 nM T39716 C53ENH 137640507 IC50 = 1300 nM T39716 CN1RV9 137640762 IC50 = 162 nM T39716 CU0BS2 137641410 IC50 = 916 nM T39716 C70XZQ 137643636 IC50 > 30000 nM T39716 C2FOK7 137644816 IC50 = 1500 nM T39716 C5UL6D 137645197 IC50 = 1900 nM T39716 CNB72K 137645644 IC50 = 415 nM T39716 CH0TP2 137645931 IC50 = 3400 nM T39716 CMG27C 137645959 IC50 = 1600 nM T39716 CDCH19 137646766 IC50 = 242 nM T39716 CFKR53 137646837 IC50 > 30000 nM T39716 C4XVD2 137647076 IC50 = 660 nM T39716 CE57QM 137647529 IC50 = 281 nM T39716 C9L8CZ 137647771 IC50 = 1900 nM T39716 CD2WA1 137647899 IC50 = 2700 nM T39716 CTD69B 137647980 IC50 = 40000 nM T39716 CL06NY 137648464 IC50 > 30000 nM T39716 C3VO8H 137648536 IC50 = 6800 nM T39716 CP32AR 137648836 IC50 = 266 nM T39716 CQ93EC 137649075 IC50 = 400 nM T39716 COLY80 137649218 IC50 > 30000 nM T39716 CUFO39 137649223 IC50 > 30000 nM T39716 CV03MT 137649269 IC50 = 520 nM T39716 CJ59RF 137649283 IC50 = 820 nM T39716 CYU2J5 137649494 IC50 = 221 nM T39716 C04JSE 137649716 IC50 > 10000 nM T39716 C6PL9C 137651460 IC50 = 430 nM T39716 CE1OC6 137651969 IC50 = 18 nM T39716 CV4AP0 137652684 IC50 = 3200 nM T39716 C65XKJ 137653127 IC50 > 30000 nM T39716 CM1CP2 137653473 IC50 = 13000 nM T39716 CMJ0X9 137654527 IC50 = 24200 nM T39716 C8BDX5 137655281 IC50 > 30000 nM T39716 C9PJC3 137655604 IC50 > 10000 nM T39716 C3LG7W 137655838 IC50 > 30000 nM T39716 CJ7D8K 137655914 IC50 = 151 nM T39716 CTW5P4 137656265 IC50 = 328 nM T39716 CN2UE9 137656598 IC50 > 30000 nM T39716 CU28CY 137657424 IC50 = 52 nM T39716 C2ME3D 137657693 IC50 > 10000 nM T39716 CA72YP 137658615 IC50 = 220 nM T39716 CDO4F5 137658625 IC50 = 1100 nM T39716 C9VOB4 137658779 IC50 = 348 nM T39716 CZ2G4H 137659479 IC50 > 30000 nM T39716 C8UK1W 137659739 IC50 = 2400 nM T39716 CH4M3X 137659806 IC50 = 94 nM T39716 C2KX3V 137661020 IC50 = 17300 nM T39716 CF8HN9 137661762 IC50 = 1400 nM T39716 C0XCS4 137661956 IC50 = 77 nM T39716 CFC3L4 137662114 IC50 = 796 nM T39716 CC9K8L 137796790 IC50 = 22000 nM T39716 C7TAV3 138319685 IC50 > 300000 nM T39716 CE79SV 138377584 IC50 > 15000 nM T39716 C81ILP 138471783 IC50 > 30000 nM T39716 CJ68PM 138558077 IC50 > 30000 nM T39716 CF78ZM 138571094 IC50 = 19000 nM T39716 CR23HX 145948497 IC50 = 25000 nM T39716 CNSU46 145948687 IC50 > 5000 nM T39716 CRH94T 145948711 IC50 > 5000 nM T39716 CDZK19 145948712 IC50 > 5000 nM T39716 C8KW9F 145948730 IC50 = 2700 nM T39716 CQPL31 145948977 IC50 > 5000 nM T39716 CF6L8Q 145955101 IC50 = 260 nM T39716 CWJ0K6 145955642 IC50 > 100000 nM T39716 CCTB54 145958837 IC50 = 6640 nM T39716 C38DYW 145959291 IC50 = 3072 nM T39716 C3PA1D 145960602 IC50 = 4000 nM T39716 CZ8W1F 145960626 IC50 > 30000 nM T39716 CX3VH5 145960676 IC50 = 27000 nM T39716 CJ1O5H 145961103 IC50 > 30000 nM T39716 CBHA12 145961383 IC50 = 1100 nM T39716 CTVR05 145961491 IC50 = 18000 nM T39716 CSAR89 145961545 IC50 = 5300 nM T39716 C90GVK 145961619 IC50 = 13000 nM T39716 CRYN14 145961777 IC50 > 30000 nM T39716 CKM9A7 145961840 IC50 > 100000 nM T39716 CIM9O6 145961922 IC50 > 100000 nM T39716 CRQ9Z2 145962160 IC50 = 10000 nM T39716 C5HE2I 145962668 IC50 = 12000 nM T39716 CWL65X 145962677 IC50 = 2600 nM T39716 C52VFR 145962752 IC50 = 1300 nM T39716 C5E3RJ 145962891 IC50 > 100000 nM T39716 C6VNH3 145962956 IC50 > 100000 nM T39716 CS86IX 145963060 IC50 = 29000 nM T39716 C8CQX3 145963143 IC50 > 100000 nM T39716 CC1T5Z 145963172 IC50 > 100000 nM T39716 CP9TU4 145963182 IC50 = 7300 nM T39716 CWS86L 145963466 IC50 = 29000 nM T39716 CF7K5G 145963483 IC50 > 30000 nM T39716 C3UZX8 145963617 IC50 = 1800 nM T39716 CB9S3T 145963706 IC50 > 100000 nM T39716 CQT0L8 145963819 IC50 = 4800 nM T39716 C91CMS 145964520 IC50 = 4400 nM T39716 CW21LJ 145964527 IC50 > 30000 nM T39716 C5MJ1S 145964650 IC50 > 30000 nM T39716 CONK20 145964797 IC50 > 30000 nM T39716 CSK8Y1 145965486 IC50 = 4020 nM T39716 C3RYM4 145965521 IC50 > 30000 nM T39716 CR1U5T 145965937 IC50 > 30000 nM T39716 CL0UK1 145966092 IC50 > 30000 nM T39716 CYB3D7 145967129 IC50 = 1700 nM T39716 CHF13C 145967515 IC50 > 30000 nM T39716 CK7PN3 145969142 IC50 = 6000 nM T39716 C05NCW 145969596 IC50 > 30000 nM T39716 C4O5HA 145972742 IC50 > 30000 nM T39716 C8RFM3 145973261 IC50 > 33000 nM T39716 C1EH5C 145975024 IC50 > 30000 nM T39716 CT6Q3V 145975287 IC50 > 30000 nM T39716 CC49BG 145975892 IC50 = 1000 nM T39716 C59HVM 145977053 IC50 > 30000 nM T39716 CC1EP9 145977316 IC50 = 5000 nM T39716 CN9Q2I 145977501 IC50 = 5600 nM T39716 CUV49K 145977796 IC50 > 10000 nM T39716 C07URC 145978291 IC50 > 30000 nM T39716 C4O0KS 145978491 IC50 > 30000 nM T39716 C3QB6J 145978986 IC50 = 2400 nM T39716 CUXB52 145979881 IC50 = 6500 nM T39716 C87TKG 145980518 IC50 = 3000 nM T39716 C7XK3P 145981121 IC50 = 10000 nM T39716 CY8IF4 145981627 IC50 > 10000 nM T39716 C8RA5D 145981858 IC50 = 27000 nM T39716 C1YW4D 145982684 IC50 = 950 nM T39716 CBK7Z6 145986895 IC50 = 7900 nM T39716 C4GA2N 145987154 IC50 = 9100 nM T39716 CNL1W0 145987554 IC50 = 4200 nM T39716 C8Q2EG 145988110 IC50 = 4870 nM T39716 CP21ZQ 145988400 IC50 = 14000 nM T39716 CP45ZX 145988718 IC50 > 42000 nM T39716 C6U7LS 145990658 IC50 = 9500 nM T39716 C42YMJ 145990677 IC50 = 9600 nM T39716 CHZB80 145990751 IC50 = 710 nM T39716 CU0K2Y 145990810 IC50 > 10000 nM T39716 CGP61R 145991617 IC50 = 140 nM T39716 C0E2AZ 145991842 IC50 = 500 nM T39716 CMP27V 145992366 IC50 = 400 nM T39716 CQY2K6 145992782 IC50 = 42000 nM T39716 CDG51F 145993858 IC50 = 11000 nM T39716 CN86HU 145994027 IC50 = 6700 nM T39716 CW3B0G 145994131 IC50 = 3100 nM T39716 CBLA80 146683623 IC50 = 4600 nM T39716 C6Q2PL 155511032 IC50 = 13000 nM T39716 CNJ74U 155511848 IC50 > 30000 nM T39716 C3LFE7 155512957 IC50 > 30000 nM T39716 CXAL69 155513487 IC50 > 30000 nM T39716 C30OPH 155516574 IC50 = 6700 nM T39716 C8DA2L 155516676 IC50 = 23000 nM T39716 C4W6SR 155517129 IC50 = 9500 nM T39716 CY5UE9 155517299 IC50 > 42000 nM T39716 C03QEN 155519060 IC50 = 8400 nM T39716 CM96HX 155520010 IC50 = 6400 nM T39716 CAG7J0 155521246 IC50 > 30000 nM T39716 C76JKY 155521282 IC50 > 30000 nM T39716 C3A1YG 155522007 IC50 > 30000 nM T39716 C26JPN 155523322 IC50 = 12000 nM T39716 COZ54G 155523716 IC50 > 10000 nM T39716 C65NKP 155524061 IC50 > 30000 nM T39716 CTM01D 155525057 IC50 > 30000 nM T39716 C9RQ1Z 155526268 IC50 = 2400 nM T39716 CZX19C 155526353 IC50 = 3100 nM T39716 CF12TX 155527767 IC50 = 11000 nM T39716 CRE0O6 155528016 IC50 = 18000 nM T39716 C5P0YG 155529298 IC50 > 30000 nM T39716 C9U8FN 155529326 IC50 = 8700 nM T39716 C4PR0S 155530319 IC50 > 30000 nM T39716 CQ15KS 155530714 IC50 = 460 nM T39716 CGO81N 155532622 IC50 = 24000 nM T39716 CZ3F2O 155533245 IC50 > 30000 nM T39716 CQE8Y5 155534372 IC50 = 5200 nM T39716 CIKQ03 155534824 IC50 = 24000 nM T39716 CXA95Z 155535618 IC50 > 30000 nM T39716 C87RFO 155536189 IC50 > 30000 nM T39716 CO71LS 155536843 IC50 > 30000 nM T39716 CG8I5F 155538033 IC50 = 19000 nM T39716 CSDO95 155538523 IC50 > 30000 nM T39716 C64QKD 155538732 IC50 > 10000 nM T39716 CW1D7Y 155538889 IC50 = 5400 nM T39716 CRQW26 155539819 IC50 > 30000 nM T39716 CH63BD 155540878 IC50 > 42000 nM T39716 CQO68V 155541113 IC50 > 30000 nM T39716 C5T9KE 155542416 IC50 > 30000 nM T39716 CEL05R 155543885 IC50 > 25000 nM T39716 CQ7W0S 155544240 IC50 > 30000 nM T39716 C9H1RS 155545131 IC50 = 16000 nM T39716 CZ47YD 155545889 IC50 = 8900 nM T39716 CPD1B3 155547824 IC50 > 30000 nM T39716 CI94QY 155550095 IC50 = 3700 nM T39716 C1WTQ7 155553777 IC50 > 30000 nM T39716 CAV3Q9 155553847 IC50 > 30000 nM T39716 C8Q2FG 155555556 IC50 = 12290 nM T39716 CGE76T 155555738 IC50 > 30000 nM T39716 C3WT2Q 155556441 IC50 > 30000 nM T39716 CJX1Q7 155557620 IC50 = 9300 nM T39716 C0T6WM 155558045 IC50 > 42000 nM T39716 CKZT21 155559364 IC50 > 33000 nM T39716 CZ0VL5 155559622 IC50 > 30000 nM T39716 CY06UB 155561401 IC50 = 21000 nM T39716 CL96XW 155562578 IC50 > 30000 nM T39716 CPL2D9 155562982 IC50 = 11600 nM T39716 CSDR68 155563772 IC50 = 4100 nM T39716 CC5FE7 155564581 IC50 > 30000 nM T39716 CJL8Y5 155565696 IC50 = 14400 nM T39716 C2EKM7 155566527 IC50 = 5900 nM T39716 CZ9OW6 155567417 IC50 > 30000 nM T39716 CE3H4Z 155567528 IC50 = 800 nM T39716 CG97KZ 155568180 IC50 = 17800 nM T39716 D00TGC 56951318 IC50 = 200 nM T39716 D01AGR 24857857 IC50 = 4600 nM T39716 D06GQO 10955473 IC50 = 9000 nM T39716 D0FF6S 16038374 IC50 = 7340 nM T39716 D0N2KU 44517677 IC50 > 26000 nM T39716 D0O2RN 22149251 IC50 = 5650 nM T39716 D0P8TL 56947150 IC50 = 210 nM T05090 D00SQN 12136798 IC50 = 265 nM T05090 D07POC 176870 IC50 > 32000 nM T05090 D08CDI 208908 IC50 > 10000 nM T05090 D09DHY 6167 IC50 > 20 ug.mL-1 T05090 D0E3SH 6918837 Ki = 1.1 nM T05090 D0E7PQ 5311 IC50 = 1.4 nM T05090 D0L7LC 5352062 Ki = 0.15 nM T05090 D0Y3KG 3121 IC50 = 161000 nM T05090 D00FHR 9865515 Ki = 265 nM T05090 D05KED 53340666 IC50 = 51 nM T05090 D06TKI 49857317 IC50 = 7 nM T05090 D07FPY 6918877 Ki = 12 nM T05090 D09XIZ 11538455 Ki = 2.1 nM T05090 D0B3FV 6445533 IC50 = 0.4 nM T05090 D0B7CH 4775 IC50 = 260000 nM T05090 D0E6UZ 54575456 IC50 = 1.8 nM T05090 D0GE5B 56654642 IC50 = 60 nM T05090 D0GH3Q 9804992 Ki = 3 nM T05090 D0L2UQ 49855250 Ki = 19 nM T05090 D0M8FD 4261 IC50 < 300 nM T05090 D0V0SL 11749858 Ki = 8.2 nM T05090 D0XT6W 6918638 Ki = 1.5 nM T05090 D0Z4RC 24756910 IC50 = 9.1 nM T05090 D03SZR 5353484 IC50 = 70 nM T05090 D0J8OC 5186 Ki = 4.1 nM T05090 D0CH8Q 56965342 IC50 = 16 nM T05090 D0N2DK 72710871 IC50 = 2 nM T05090 D0QX3G 71532921 IC50 = 1700 nM T05090 D0N3SH 4996 Ki = 8 nM T05090 D0W9NH 2746 IC50 = 46 nM T05090 CBIR94 10313 IC50 = 7830 nM T05090 CL25FN 76175 IC50 > 30000 nM T05090 C1N2KZ 88129 IC50 = 340000 nM T05090 CH1JD3 419176 IC50 = 10000 nM T05090 CU3HS2 1108280 IC50 > 100000 nM T05090 C18ENP 6918846 Ki = 11 nM T05090 C1RD7E 6918878 IC50 = 398 nM T05090 CE9LP2 9543539 IC50 = 69 nM T05090 CJ07ZA 9800555 IC50 = 67 nM T05090 CC0EU7 9828788 IC50 = 4.8 nM T05090 C81EYJ 9923508 IC50 = 4.9 nM T05090 CQG4V8 9924543 IC50 = 2.8 nM T05090 CZL7C8 10017099 IC50 = 10 nM T05090 CL4C9H 10154438 Ki = 2.7 nM T05090 C7RC1E 10309899 IC50 = 9 nM T05090 C8G5WP 11210533 IC50 = 6900 nM T05090 CYJ60V 11244651 IC50 = 80100 nM T05090 CY34EQ 11393847 IC50 > 20000 nM T05090 CRZ7H2 11556677 IC50 = 12 nM T05090 C24SBP 11657529 IC50 = 250 nM T05090 CQ32FV 11664499 IC50 = 1.6 nM T05090 CG9OC4 11682502 IC50 = 30 nM T05090 CYB26W 11688197 IC50 = 187 nM T05090 CC3GQ0 11700059 IC50 = 48 nM T05090 C9G1BN 11993595 IC50 = 440 nM T05090 CH5JS7 11993694 IC50 = 23 nM T05090 C1BVY9 12325934 IC50 > 30000 nM T05090 C06UTF 13507024 IC50 = 10 nM T05090 C4XJ8M 13889849 Ki = 1350 nM T05090 C1KR4L 14113324 IC50 > 50000 nM T05090 C15MQN 14113325 IC50 > 50000 nM T05090 C2D1KP 15983982 Ki = 20 nM T05090 CA2YF9 15984018 IC50 = 230 nM T05090 CB81VC 15985904 IC50 = 130 nM T05090 CHB82E 15986417 IC50 = 55600 nM T05090 C52EVH 15986418 IC50 = 4570 nM T05090 CS1QO9 15986509 IC50 = 84500 nM T05090 C5T1WF 16006672 IC50 = 697 nM T05090 CQGC05 16036765 IC50 = 14 nM T05090 CM3T2E 16049824 IC50 = 17 nM T05090 C30UFT 16066811 IC50 = 939 nM T05090 CFK8J5 16068056 Ki = 20 nM T05090 CMQP70 16068495 Ki = 27 nM T05090 CT84XO 16068594 Ki = 15 nM T05090 CF3ZG5 16068595 Ki = 13 nM T05090 CL60CA 16068912 Ki = 10 nM T05090 CVT0E7 16070046 IC50 = 276 nM T05090 C5CIB4 16663079 IC50 > 50000 nM T05090 CWO7V0 16733295 IC50 = 1560 nM T05090 CV54SY 16733414 IC50 = 1320 nM T05090 CB4IN2 16773791 IC50 = 289 nM T05090 CKM7F9 17747371 IC50 > 1000 nM T05090 CF7JR0 17756401 IC50 = 50 nM T05090 C3FN8M 17756403 IC50 = 79 nM T05090 CE2W3M 21630365 IC50 = 988 nM T05090 CS5R0U 22836624 Ki = 14500 nM T05090 CEF8W4 23625604 IC50 = 3162.28 nM T05090 CB8A5Q 23648260 IC50 = 27710 nM T05090 C36NKL 23648268 IC50 > 20000 nM T05090 C4UV3T 24726843 IC50 = 3500 nM T05090 C8RC9P 24744325 IC50 = 7000 nM T05090 CMI5E4 24746277 IC50 = 16480 nM T05090 CVB7J3 24746434 IC50 = 1260000 nM T05090 C8EYH1 24746435 IC50 = 340000 nM T05090 C28AWJ 24746436 IC50 = 1270000 nM T05090 C17GDO 24779722 IC50 = 131 nM T05090 CIO7Q6 24853792 IC50 = 1000 nM T05090 CBN0J5 24853793 IC50 = 120 nM T05090 CI3B6L 24857909 IC50 = 670 nM T05090 C5GCM1 24881328 IC50 = 13.7 nM T05090 C8QVB1 24881329 IC50 = 25.3 nM T05090 CU0AM3 24881330 IC50 = 7.9 nM T05090 CQM51L 24881331 IC50 = 7.2 nM T05090 C4KH8F 24881332 IC50 = 16.4 nM T05090 C1KA3V 24881333 IC50 = 15.1 nM T05090 C47APB 24881402 IC50 = 4.5 nM T05090 CSN8W1 24881403 IC50 = 7.7 nM T05090 C1UQ3K 24881404 IC50 = 8 nM T05090 C51TMH 24881405 IC50 = 4 nM T05090 C9EZI7 24881406 IC50 = 2.7 nM T05090 C6P3HS 24881407 IC50 = 9.7 nM T05090 CZ3TU1 24881464 IC50 = 12 nM T05090 CDI49N 24881465 IC50 = 5.8 nM T05090 CQGP87 24881466 IC50 = 4.2 nM T05090 CS1MH8 24888322 IC50 = 22000 nM T05090 CC0R9O 24938735 IC50 = 0.7 nM T05090 CF03HD 24948905 IC50 = 115 nM T05090 CHP8O6 24948906 IC50 = 4.04 nM T05090 C1KRT8 24948907 IC50 = 144 nM T05090 CKY2P8 24948908 IC50 = 10.2 nM T05090 C25CFI 24948909 IC50 = 65.8 nM T05090 CWQ04Z 24948910 IC50 = 18 nM T05090 CM9I3X 24951310 IC50 = 12.9 nM T05090 CX1YF8 24951311 IC50 = 158 nM T05090 CV10XU 24951312 IC50 < 0.002 nM T05090 CD6KV0 24951313 IC50 = 83.6 nM T05090 CQY9Z0 24951314 IC50 = 190 nM T05090 C5B0IJ 25023793 IC50 = 120 nM T05090 CLG23N 25023794 IC50 = 10 nM T05090 CHE82I 25023795 IC50 > 10000 nM T05090 CX8G3W 25023796 IC50 = 1700 nM T05090 CVRS37 25023797 IC50 = 560 nM T05090 C7GO3U 25023798 IC50 = 9400 nM T05090 C3G2AU 25023799 IC50 = 120 nM T05090 CAS18V 25023800 IC50 = 3100 nM T05090 CX7D5B 25023801 IC50 = 1400 nM T05090 CZG50I 25023802 IC50 > 5000 nM T05090 CP4T7J 25023806 IC50 = 2900 nM T05090 CVS1M4 25023811 IC50 = 4600 nM T05090 CJG8C5 25023818 IC50 = 7300 nM T05090 CLA50V 25023819 IC50 = 7600 nM T05090 CV8EF6 25032862 IC50 = 22450 nM T05090 CX69SY 25066355 IC50 = 369 nM T05090 CF8VP4 25066356 IC50 = 176 nM T05090 CS9XH7 25066547 IC50 = 240 nM T05090 C46AGN 25066548 IC50 = 39.6 nM T05090 CJF2M7 25066549 IC50 = 246 nM T05090 CPTI96 25110599 IC50 = 12 nM T05090 C7ZN2W 25118059 IC50 = 3.4 nM T05090 C4I1CJ 25155417 IC50 = 6180 nM T05090 CB4E2J 25155956 IC50 > 50000 nM T05090 CKG24O 25157972 IC50 = 6390 nM T05090 C19JIO 25157973 IC50 = 5384 nM T05090 CFS5O4 25168576 IC50 = 7100 nM T05090 C0R5OK 25168856 IC50 > 1000 nM T05090 CO14XG 25195084 IC50 = 320 nM T05090 C6BDX3 25207860 IC50 = 104000 nM T05090 C5COM1 25218554 IC50 = 6928 nM T05090 CN6XA4 25218555 IC50 = 9617 nM T05090 CL8K9U 25218556 IC50 = 8706 nM T05090 C9WA4B 25218557 IC50 = 17390 nM T05090 CRG29Y 25218558 IC50 = 5727 nM T05090 CEH71M 25218560 IC50 = 4330 nM T05090 CIZD97 25218561 IC50 > 50000 nM T05090 C7I5EL 25218562 IC50 = 3202 nM T05090 C15YDI 25218563 IC50 = 5102 nM T05090 CCD5M7 25227504 IC50 = 55.7 nM T05090 CK0D5S 25227505 IC50 = 89 nM T05090 CN97JP 25227508 IC50 = 93.6 nM T05090 CW8R1B 25227513 IC50 = 94.5 nM T05090 CPNQ02 25257992 IC50 = 85 nM T05090 CE0NV4 25257993 IC50 = 3.07 nM T05090 C43BHY 25269097 IC50 = 25 nM T05090 CU53WB 42596953 IC50 = 66 nM T05090 C2LES7 42599455 IC50 = 5.3 nM T05090 C2KO0F 42599456 IC50 = 6.7 nM T05090 C1UAO7 42601485 IC50 = 12000 nM T05090 COI7Y3 42611300 IC50 = 143 nM T05090 CU23PG 42611301 IC50 = 8 nM T05090 CW1G2R 42611390 IC50 = 280 nM T05090 CQ37HN 42612743 IC50 = 2.59 nM T05090 CX1UT9 42612744 IC50 = 1151 nM T05090 CLH2Q7 42612852 IC50 = 608 nM T05090 CXK4C1 42618298 IC50 = 1.2 nM T05090 CDT65Y 42631047 IC50 > 100000 nM T05090 CO57GS 44138033 IC50 = 659 nM T05090 C7RCY4 44178890 IC50 = 9 nM T05090 CQ2VD5 44219634 IC50 = 25 nM T05090 C0JY2Q 44249789 IC50 = 1300 nM T05090 CU7SL0 44249820 IC50 = 2200 nM T05090 CY0QB9 44253226 IC50 = 65 nM T05090 CZ8R1N 44253780 IC50 = 87 nM T05090 C5YRC9 44431499 IC50 = 91000 nM T05090 CV7P0C 44447120 IC50 = 2810 nM T05090 CNC51G 44447194 IC50 > 50000 nM T05090 C8WKU9 44453790 IC50 = 42 nM T05090 C5VP4D 44454144 IC50 = 11000 nM T05090 C8A1ZD 44456564 IC50 = 3.7 nM T05090 CJ0L4C 44456965 IC50 = 14 nM T05090 C74LTB 44506448 IC50 = 61 nM T05090 C4FKU6 44541235 IC50 > 1000 nM T05090 C7F8YJ 44543715 Ki = 250 nM T05090 CQ2TU3 44550557 Ki = 740 nM T05090 CW4KH2 44551271 IC50 = 16800 nM T05090 CDW54Z 44562605 IC50 > 1000 nM T05090 C9MB4K 44562607 IC50 = 500 nM T05090 CH2NP3 44562608 IC50 > 1000 nM T05090 CBYZ26 44562609 IC50 > 1000 nM T05090 C3QSI4 44562762 IC50 > 1000 nM T05090 CRJS52 44562763 IC50 > 1000 nM T05090 CJ5US8 44562765 IC50 > 1000 nM T05090 CQ5RJ3 44562799 IC50 = 630 nM T05090 CDY0E1 44562801 IC50 > 1000 nM T05090 CEM91G 44562802 IC50 = 380 nM T05090 CEA9D0 44562840 IC50 > 1000 nM T05090 C3DMN0 44563197 IC50 = 520 nM T05090 CGF8R5 44563236 IC50 > 1000 nM T05090 CT63QG 44563237 IC50 = 500 nM T05090 CIO34V 44564642 Ki = 11 nM T05090 COM65J 44572384 IC50 = 620 nM T05090 CMA3R6 44574139 IC50 = 30 nM T05090 C5KLR7 44574177 IC50 > 30000 nM T05090 CFS49I 44574178 IC50 = 10600 nM T05090 CJ32DK 44574179 IC50 > 30000 nM T05090 CQOS28 44574180 IC50 = 102 nM T05090 CN96ZV 44574181 IC50 = 7410 nM T05090 C46XHW 44574207 IC50 > 30000 nM T05090 C3RY9V 44574208 IC50 = 1920 nM T05090 CS4JP5 44589733 IC50 > 10000 nM T05090 CEPG12 44589734 IC50 = 840 nM T05090 CZVO54 44589735 IC50 = 1500 nM T05090 CPB1G7 44589736 IC50 = 2800 nM T05090 CZ7VE6 44589745 IC50 = 27 nM T05090 CDH14U 44589746 IC50 = 180 nM T05090 C3C6WU 44589911 IC50 = 5340000 nM T05090 CVA4I9 44589912 IC50 = 5500000 nM T05090 CVQ83W 44589913 IC50 > 30000000 nM T05090 C16-FEB 44591258 IC50 = 19320 nM T05090 C1OCI9 44591315 IC50 = 4803 nM T05090 CA6Q9Y 44592060 IC50 = 3140 nM T05090 CH2J8R 44598238 IC50 = 1670 nM T05090 CE5W3U 44598288 IC50 = 690 nM T05090 C68BJH 44598289 IC50 = 2990 nM T05090 C9K2WV 44598290 IC50 = 970 nM T05090 C16ZEP 44598291 IC50 = 54 nM T05090 C28GHB 44598344 IC50 = 260 nM T05090 CU65LR 44598345 IC50 = 262 nM T05090 C41VTN 44598346 IC50 = 1090 nM T05090 CHQ86X 44598347 IC50 = 694 nM T05090 CCVA51 44598385 IC50 = 1040 nM T05090 C29NXL 44598386 IC50 = 3630 nM T05090 C5WM7H 44598387 IC50 > 10000 nM T05090 CK8V9I 44598388 IC50 = 164 nM T05090 CJ54OH 44598429 IC50 = 31 nM T05090 C1TYW6 44598430 IC50 = 240 nM T05090 C3TOK2 44598431 IC50 = 190 nM T05090 CPZ65Q 44598479 IC50 > 10000 nM T05090 CGT51H 44598480 IC50 = 62 nM T05090 CZ62IW 44598481 IC50 > 10000 nM T05090 C0OT6I 44598482 IC50 = 7080 nM T05090 CX8U6S 44598483 IC50 > 10000 nM T05090 CO5YJ8 44598535 IC50 = 990 nM T05090 C5H8RA 44598536 IC50 = 32 nM T05090 CC2QV9 44623002 IC50 > 50000 nM T05090 CVJ51M 44623152 IC50 > 50000 nM T05090 C6TJ2G 44623153 IC50 > 50000 nM T05090 COZ25S 45268021 IC50 = 69300 nM T05090 CS9DW4 45268025 IC50 = 3400 nM T05090 C0BQF9 45268900 IC50 = 46900 nM T05090 CH08UF 45268906 IC50 = 5600 nM T05090 C27VLQ 45269750 IC50 = 4300 nM T05090 CK1AP8 45269751 IC50 = 27200 nM T05090 CSM1O6 45271073 IC50 = 260 nM T05090 C02LVF 45485792 IC50 = 32 nM T05090 C7EAV5 45485820 IC50 = 54 nM T05090 CIO0T2 46179730 IC50 = 3.39 nM T05090 C2M4GV 46179732 IC50 = 3.7 nM T05090 CS75CD 46179779 IC50 = 2.8 nM T05090 C39YKM 46179780 IC50 = 5.3 nM T05090 C0CKE5 46180624 IC50 = 120 nM T05090 C7GYH0 46180758 IC50 = 18.1 nM T05090 C27IKH 46180759 IC50 = 3 nM T05090 CSC1Y9 46180760 IC50 = 3.4 nM T05090 C4XHL5 46180761 IC50 = 1.4 nM T05090 C70FSJ 46180763 IC50 = 3.3 nM T05090 CD57RJ 46197798 IC50 = 9 nM T05090 CR04HA 46197799 IC50 = 21 nM T05090 CB2G1W 46881144 IC50 = 1.66 nM T05090 C85RDN 46881213 IC50 = 1.55 nM T05090 CQTI31 46881225 IC50 = 122 nM T05090 C48QWG 46884058 IC50 = 2263 nM T05090 CVU0D3 46884059 IC50 = 35 nM T05090 C5UMJ3 46884060 IC50 = 240 nM T05090 CQ76JG 46884061 IC50 = 1750 nM T05090 C9HMN4 46884114 IC50 = 1100 nM T05090 C8V3HK 46884115 IC50 = 1346 nM T05090 C8CI2D 46884116 IC50 = 4989 nM T05090 C35OPR 46884117 IC50 = 56 nM T05090 CI0W9C 46884118 IC50 = 30 nM T05090 C25DSY 46887918 IC50 = 24.7 nM T05090 C93CLK 46887919 IC50 = 22000 nM T05090 CPSI47 46890583 Ki = 8 nM T05090 C90NYX 46896338 IC50 = 230 nM T05090 CU7L5W 46906597 IC50 = 470000 nM T05090 CG46KJ 46906641 IC50 = 605000 nM T05090 CAT34L 46906643 IC50 = 36000 nM T05090 C4V7PG 46907052 IC50 = 13300 nM T05090 CSNU34 46907053 IC50 = 3200 nM T05090 CMQ3R0 46907054 IC50 = 14500 nM T05090 C05KTS 46907124 IC50 = 460000 nM T05090 C2PC1Z 46907160 IC50 = 32300 nM T05090 C72BEW 46907196 IC50 = 730000 nM T05090 C4V3ZK 46907197 IC50 = 718000 nM T05090 C6TRS7 46907198 IC50 = 695000 nM T05090 C0K4DL 46907280 IC50 = 725000 nM T05090 C3NE0Q 46907281 IC50 = 508000 nM T05090 C1HV6U 46907409 IC50 > 20000 nM T05090 C6GY9I 46934544 IC50 = 26700 nM T05090 C3OD2Y 46934546 IC50 = 28100 nM T05090 CL7PS1 49831258 IC50 = 46000 nM T05090 CC7Y9U 49850262 IC50 = 155 nM T05090 C50PXU 49855444 IC50 > 50000 nM T05090 CE7D2J 49855568 IC50 = 6300 nM T05090 CFD9P3 49855569 IC50 > 32000 nM T05090 C1AU5N 49855758 IC50 > 32000 nM T05090 CIFK93 49855759 IC50 > 32000 nM T05090 CK48OJ 49855760 IC50 > 32000 nM T05090 CZI3M1 49855761 IC50 > 32000 nM T05090 CRPZ58 49855949 IC50 > 32000 nM T05090 CTU0K3 49855950 IC50 > 32000 nM T05090 CF85NL 49855951 IC50 > 32000 nM T05090 CF7YS9 49855952 IC50 > 32000 nM T05090 CJU38G 49855953 IC50 = 560 nM T05090 C6POK9 49856931 IC50 = 10 nM T05090 C52ABG 50942502 IC50 = 460 nM T05090 CPQ0F7 50991199 IC50 = 2 nM T05090 COA5W3 51051073 IC50 = 28 nM T05090 C5LZ4R 51351536 IC50 > 30000 nM T05090 CV76KB 51357270 IC50 = 30 nM T05090 C8SUQ5 53317424 IC50 > 30000 nM T05090 C7MO2J 53325871 IC50 = 2.1 nM T05090 CG84JS 53325976 IC50 = 1000 nM T05090 CVM4Q3 53357987 IC50 = 20000 nM T05090 C78GKN 53361474 Ki = 64 nM T05090 CNB63X 53361475 Ki = 23 nM T05090 CQ43VH 53363518 Ki = 16 nM T05090 C6Y2EV 53374826 IC50 = 5370 nM T05090 CC5K2U 53380601 IC50 = 760 nM T05090 CN17BX 53380699 IC50 = 1520 nM T05090 CYQV72 54030066 IC50 = 39000 nM T05090 C5A7MU 54613496 IC50 = 6.4 nM T05090 CVP16C 54753629 IC50 = 97000 nM T05090 CIO96M 56659403 IC50 > 100000 nM T05090 CT4ZY0 56661203 IC50 = 6 nM T05090 C7R9TZ 56663191 IC50 = 0.7 nM T05090 CL18NI 56666337 IC50 > 100000 nM T05090 C9LC5Y 56673234 IC50 > 100000 nM T05090 CWH5N4 56673261 IC50 > 100000 nM T05090 C2ML5S 56837168 IC50 = 9.77 nM T05090 CCW89V 56932477 IC50 = 0.669 nM T05090 CZ25SN 56935695 IC50 > 30000 nM T05090 CP4EL2 57328394 IC50 = 14000 nM T05090 C5CRJ1 57412107 IC50 = 90 nM T05090 COG4Q8 57412108 IC50 = 130 nM T05090 C4LI0D 57521296 IC50 = 4700 nM T05090 CA5Q6O 58147189 IC50 > 50000 nM T05090 C4DYC0 58147224 IC50 > 50000 nM T05090 CMP04X 58147302 IC50 > 50000 nM T05090 C4V7FY 58191950 IC50 = 840 nM T05090 CPCA29 58191961 IC50 = 15 nM T05090 C7HF1L 58191965 IC50 = 550 nM T05090 CR4BX0 58191982 IC50 = 440 nM T05090 C8V1NK 58191988 IC50 = 920 nM T05090 C8LWY9 58191997 IC50 = 510 nM T05090 C3IQ9B 58191999 IC50 = 770 nM T05090 CQB69R 58192003 IC50 = 610 nM T05090 CLD40J 58465708 IC50 = 8500 nM T05090 C1MB4Q 59323957 IC50 > 30000 nM T05090 CK6LX0 59454220 IC50 = 230 nM T05090 C2SDN1 59454252 IC50 = 200 nM T05090 CPZ5Q3 60148646 IC50 = 25000 nM T05090 CP2HK9 60148667 IC50 = 18000 nM T05090 C8ZL3J 60148690 IC50 = 16000 nM T05090 CK5N4E 60148693 IC50 = 12000 nM T05090 C27DKW 60148711 IC50 = 9400 nM T05090 CS2E6C 60148712 IC50 = 26000 nM T05090 CPF50R 60148997 IC50 = 33000 nM T05090 CB7X2E 60151224 IC50 = 7.67 nM T05090 CY05OU 60151225 IC50 = 73 nM T05090 CWO8H0 60152596 IC50 = 1680 nM T05090 CBN3L0 69950064 Ki > 43000 nM T05090 C6RFQ8 70676597 IC50 = 3000 nM T05090 CM4XB8 70681905 IC50 = 5090 nM T05090 CW5MP0 70681906 IC50 = 4890 nM T05090 CGYX13 70681907 IC50 = 5700 nM T05090 CPMZ01 70681908 IC50 = 2190 nM T05090 CM62BN 70682297 IC50 = 1440 nM T05090 C3PR4C 70684025 IC50 = 34120 nM T05090 C8R9XE 70684026 IC50 = 4800 nM T05090 CT64UC 70686159 IC50 = 16070 nM T05090 C94YFZ 70686160 IC50 = 26390 nM T05090 CBZ8W0 70688300 IC50 = 13480 nM T05090 C0CQP5 70690303 IC50 = 6620 nM T05090 C8T1FV 70690304 IC50 = 1940 nM T05090 C7VF1B 70692849 IC50 = 800 nM T05090 C28UMB 70693708 IC50 = 62 nM T05090 CGSM24 70694519 IC50 = 2660 nM T05090 CX23AC 70696578 IC50 = 9380 nM T05090 CW6F1J 70696579 IC50 = 19200 nM T05090 CQY1I6 70789579 Ki > 43000 nM T05090 C76SGF 71457594 IC50 = 5400 nM T05090 C72DJO 71465631 IC50 = 1090 nM T05090 CQ7VL0 71467493 IC50 = 60 nM T05090 C5BR1D 71467494 IC50 = 110 nM T05090 CS74UB 71467495 IC50 = 2830 nM T05090 CX3U9M 71467628 IC50 = 3560 nM T05090 C3PIK2 71467958 IC50 = 110 nM T05090 CTNS49 71467959 IC50 = 620 nM T05090 CQ6B2I 71467960 IC50 = 260 nM T05090 C0YXF2 71467961 IC50 = 360 nM T05090 C1MH5Z 71467962 IC50 = 100 nM T05090 C7ESZ2 71467963 IC50 = 190 nM T05090 C45FCJ 71468055 IC50 = 380 nM T05090 C3H0CR 71468158 IC50 = 140 nM T05090 CQ26IW 71468159 IC50 = 110 nM T05090 C6ZPJ4 71468160 IC50 = 2590 nM T05090 CJU64Z 71468161 IC50 = 73.91 nM T05090 CD8O7W 71468162 IC50 = 330 nM T05090 CSDO79 71468163 IC50 = 280 nM T05090 CN97RG 71468164 IC50 = 380 nM T05090 C5I0TX 71468273 IC50 = 310 nM T05090 CJKU04 71468274 IC50 = 450 nM T05090 CZJ84E 71468275 IC50 = 590 nM T05090 C6L0RV 71468277 IC50 = 200 nM T05090 CAH65F 71468278 IC50 = 80 nM T05090 CVP26X 71468393 IC50 = 160 nM T05090 CFW2I5 71468672 IC50 = 27.51 nM T05090 CIS73X 71468801 IC50 = 1640 nM T05090 CS86BK 71468803 IC50 = 3170 nM T05090 CJD46S 71468805 IC50 = 2220 nM T05090 CU9FQ3 71468924 IC50 = 1580 nM T05090 C01IKD 71468927 IC50 = 270 nM T05090 CNXK19 71468928 IC50 = 150 nM T05090 C7GY8U 71495390 IC50 = 69 nM T05090 CBE46I 71495482 IC50 = 81 nM T05090 CQ5FC3 71495575 IC50 = 188 nM T05090 CIQ3E7 71495576 IC50 = 155 nM T05090 CAL79Y 71495577 IC50 = 49 nM T05090 C1SXH7 71495578 IC50 = 9.6 nM T05090 C1Q8LP 71495673 IC50 = 69 nM T05090 CF72JS 71495674 IC50 = 217 nM T05090 C3T7UP 71495675 IC50 = 53 nM T05090 CSW12I 71502605 IC50 = 230 nM T05090 C89SWX 71527724 IC50 = 15000 nM T05090 C6S5JQ 71527847 IC50 = 7.5 nM T05090 C6KBD4 71534512 IC50 = 72 nM T05090 CT51EW 71534810 IC50 = 3 nM T05090 C7QN3O 71534812 IC50 = 1 nM T05090 C8M3HU 71537640 IC50 = 55 nM T05090 C2QML7 71537641 IC50 = 2 nM T05090 CZJX53 71537927 IC50 = 6330 nM T05090 CU0ZE6 71537928 IC50 = 5 nM T05090 CH9FS7 71537929 IC50 = 122 nM T05090 CTW95A 71537931 IC50 = 5 nM T05090 CW3BT5 71537932 IC50 = 17100 nM T05090 C3C0RO 71538475 IC50 = 7 nM T05090 CIA28E 71538746 IC50 = 10 nM T05090 CFCV26 71538748 IC50 = 495 nM T05090 CY2T1Q 71538749 IC50 = 475 nM T05090 C4A6VJ 71538750 IC50 = 8 nM T05090 CG72NC 71538751 IC50 = 9 nM T05090 C7RUE6 71540743 IC50 = 14000 nM T05090 C9LA4F 71540744 IC50 = 885 nM T05090 C0EK5J 71540745 IC50 = 3990 nM T05090 C80HZX 71540746 IC50 = 31 nM T05090 C5UZQ0 71540747 IC50 = 10400 nM T05090 C4G5US 71540862 IC50 = 649 nM T05090 CKR6U8 71583101 IC50 = 23000 nM T05090 CBZ5S9 71583103 IC50 = 29000 nM T05090 C3PSJ9 71583105 IC50 = 26000 nM T05090 C21GHR 71624738 IC50 = 1600 nM T05090 C7HG0K 71655802 IC50 = 694 nM T05090 CV73YD 71660259 IC50 = 1360 nM T05090 CQ5UR0 71660260 IC50 = 8360 nM T05090 CQ5P0T 71660261 IC50 = 830 nM T05090 C8EIX0 71660262 IC50 = 1030 nM T05090 CPJ4V7 71680913 IC50 = 23000 nM T05090 CI9G3B 71681069 IC50 = 18000 nM T05090 CIR56T 71721558 IC50 = 260 nM T05090 CCD18W 71721946 IC50 = 240 nM T05090 CI9H6L 72164895 IC50 = 19 nM T05090 CS5UL7 72195322 IC50 = 68 nM T05090 CAC5Q7 72375561 IC50 = 550 nM T05090 C3WQV2 72375562 IC50 = 7.2 nM T05090 CC1W6J 72375670 IC50 = 1900 nM T05090 CY8R0O 72696205 IC50 = 11620 nM T05090 CM3KS6 72696333 IC50 = 1690 nM T05090 CI2EH8 72696334 IC50 = 520 nM T05090 C0CM8Q 72696335 IC50 = 230 nM T05090 CG31RX 72696336 IC50 = 2110 nM T05090 CJ3EH7 72696464 IC50 = 590 nM T05090 C1OA0T 72696465 IC50 = 130 nM T05090 C1I9TZ 72696466 IC50 = 193 nM T05090 CFU3V5 72696467 IC50 = 242 nM T05090 CTR52Z 72696598 IC50 = 767 nM T05090 C4O2ZT 72696599 IC50 = 111 nM T05090 C5N9BQ 72696600 IC50 = 1444 nM T05090 CE87BF 72696601 IC50 = 899 nM T05090 C73XOU 72734382 IC50 = 64 nM T05090 CQA16N 72946833 IC50 = 62 nM T05090 CHQ39Y 72947043 IC50 = 88 nM T05090 CCST90 72947044 IC50 = 11 nM T05090 CX3W1T 73333311 IC50 = 4500 nM T05090 C68LBO 73349131 IC50 = 2 nM T05090 CUD02X 73355098 IC50 = 102 nM T05090 CD6L5K 73707349 IC50 = 2 nM T05090 C26KZD 73707535 IC50 = 1.4 nM T05090 CM1H3U 73707536 IC50 = 5.4 nM T05090 CH97TE 73707543 IC50 = 1.8 nM T05090 C2PWQ3 73707544 IC50 = 2.4 nM T05090 CEM5B6 73707545 IC50 = 1.6 nM T05090 CPQ43R 73707550 IC50 = 0.8 nM T05090 CJ1DA8 73774764 IC50 = 403.2 nM T05090 CQ3K6G 73776326 IC50 = 14.1 nM T05090 CC4L0G 73776327 IC50 = 143 nM T05090 CZB6G7 73776472 IC50 = 3.9 nM T05090 CSRE84 73776614 IC50 = 5.5 nM T05090 C01FVX 73776616 IC50 = 3.2 nM T05090 C3UC9H 73891099 IC50 = 12400 nM T05090 CMU19S 74221664 IC50 = 330 nM T05090 CM6H9C 76324878 IC50 = 8900 nM T05090 CKI74A 76853213 IC50 > 20000 nM T05090 CCR7L2 76853289 IC50 = 12000 nM T05090 CJ6Z0X 78324068 IC50 > 20000 nM T05090 CG5ZD9 86291495 IC50 = 15 nM T05090 C3EM7H 86581004 IC50 = 85 nM T05090 C7UK3Y 86581005 IC50 = 69 nM T05090 CY64UM 86581152 IC50 = 91 nM T05090 CY5V7C 86581153 IC50 = 89 nM T05090 C1HE8I 86581432 IC50 = 210 nM T05090 CZM07I 86581434 IC50 = 65 nM T05090 C8ZQG9 86581435 IC50 = 87 nM T05090 CS5I4Y 87261507 IC50 = 80 nM T05090 C5JIT0 87618609 IC50 = 320 nM T05090 CRQO37 88005144 IC50 = 500 nM T05090 CP1NA9 89183138 IC50 > 33330 nM T05090 CQS6C0 89183185 IC50 = 1490 nM T05090 CB47VC 89464167 IC50 = 35800 nM T05090 CD7J6C 90644927 IC50 = 200 nM T05090 C62GSL 90654859 IC50 = 47 nM T05090 CYW51P 90654946 IC50 = 340000 nM T05090 CJH1S6 90654947 IC50 > 100000 nM T05090 CSDO81 90664458 Ki = 19 nM T05090 CAQL21 91667420 IC50 = 42.5 nM T05090 C5M9AK 91667421 IC50 = 14.59 nM T05090 CJO6T1 91810840 IC50 = 2100 nM T05090 CYJ12Q 91884636 IC50 = 5 nM T05090 C0FCU9 91938063 IC50 = 25.84 nM T05090 C34WIG 92045024 IC50 > 100000 nM T05090 CYO9J5 101879983 IC50 = 3.56 nM T05090 C9OC0F 101882265 IC50 = 6590 nM T05090 CVE07R 101882857 IC50 = 394 nM T05090 C63EWT 101882858 IC50 = 2.42 nM T05090 C8KZB4 101883993 Ki = 800 nM T05090 C7Q6ID 101884982 IC50 = 13 nM T05090 CR46PQ 101884983 IC50 = 6 nM T05090 CRZ83C 101884989 IC50 = 138 nM T05090 CS2UL0 117829456 IC50 = 28 nM T05090 C7L4OT 117829461 IC50 = 28 nM T05090 C50VUN 117829462 IC50 = 98 nM T05090 CH27PR 118613747 IC50 = 7.8 nM T05090 C0OX4M 118613748 IC50 = 1.1 nM T05090 CNF09H 118613750 IC50 = 100 nM T05090 C3ETI2 118613751 IC50 = 4.2 nM T05090 C9KZQ0 118613755 IC50 = 1.1 nM T05090 C30OPU 118613756 IC50 = 6 nM T05090 C46TFD 118613757 IC50 = 1.8 nM T05090 C1J5AG 118613783 IC50 = 0.68 nM T05090 C9T0ML 118613821 IC50 = 0.38 nM T05090 CSU52M 118656852 IC50 = 24000 nM T05090 C45UYG 118709095 IC50 = 12000 nM T05090 C7QHE4 118712502 IC50 = 0.3 nM T05090 C8KSD6 118712503 IC50 = 0.6 nM T05090 C1JFZ7 118714371 IC50 = 367 nM T05090 CXF0U3 118714375 IC50 = 246 nM T05090 C2M5OR 118714376 IC50 = 13 nM T05090 CY4GN9 118714377 IC50 = 30 nM T05090 C7P3KH 118715726 IC50 = 126.56 nM T05090 CK6UM0 118715727 IC50 = 37.67 nM T05090 CW85VZ 118715728 IC50 = 17.91 nM T05090 C39EXL 118715729 IC50 = 607.03 nM T05090 CYGT73 118715730 IC50 = 48.26 nM T05090 CCAM49 118715731 IC50 = 23.53 nM T05090 C37NXA 118715732 IC50 = 16.85 nM T05090 CEN1J3 118715733 IC50 = 14.47 nM T05090 CFD2B8 118715734 IC50 = 11.88 nM T05090 CO8TJ6 118715735 IC50 = 13.52 nM T05090 C90TIX 118715736 IC50 = 14.63 nM T05090 C14KQU 118715737 IC50 = 6.46 nM T05090 CMK8B7 118715738 IC50 = 20.77 nM T05090 CQ6V9M 118715739 IC50 = 3.47 nM T05090 CWM04T 118715740 IC50 = 9.33 nM T05090 CLYS39 118715741 IC50 = 2.92 nM T05090 C04XZU 118715742 IC50 = 14.74 nM T05090 CJ4FS3 118715743 IC50 = 39.72 nM T05090 C3BH1K 118715744 IC50 = 3.52 nM T05090 CA12OP 118715745 IC50 = 3.22 nM T05090 C51RTI 118715746 IC50 = 3.58 nM T05090 CFX16A 118715747 IC50 = 8.19 nM T05090 C5OWL1 118715748 IC50 = 14.05 nM T05090 C8AW9X 118715749 IC50 = 14.1 nM T05090 C2Y7ZC 118715750 IC50 = 26.53 nM T05090 CM5QT7 118719376 Ki = 1400 nM T05090 CPB7C3 118719377 Ki = 500 nM T05090 C09OGH 118719378 Ki = 600 nM T05090 CR5VC1 118719379 Ki = 700 nM T05090 C32LCM 118719380 Ki = 200 nM T05090 C8U6YR 118719381 Ki = 500 nM T05090 C9Y0HV 118719382 Ki = 300 nM T05090 CY0J4D 118719383 Ki = 500 nM T05090 CCYU59 118719817 IC50 = 11 nM T05090 CSC47W 118720522 IC50 = 223.6 nM T05090 CUI51W 118720529 IC50 = 28.7 nM T05090 CMV2W9 118721625 IC50 = 3 nM T05090 CF5TO3 118721859 IC50 = 49 nM T05090 CK97TZ 118721860 IC50 = 4 nM T05090 CYV30O 118721861 IC50 = 3 nM T05090 C5WYI1 118721862 IC50 = 5 nM T05090 CSMW25 118721863 IC50 = 897 nM T05090 C5B1KM 118721864 IC50 = 98 nM T05090 CG8LZ0 118721865 IC50 = 2710 nM T05090 CPCN23 118721866 IC50 = 2950 nM T05090 CM0A9U 118721867 IC50 = 2600 nM T05090 C8IAG9 118734664 IC50 = 12100 nM T05090 CJ6KL7 118734665 IC50 = 1970 nM T05090 C2VQ5P 118734666 IC50 = 10780 nM T05090 CYF71E 118734667 IC50 = 1490 nM T05090 CQC7H0 118734668 IC50 = 11230 nM T05090 CP27CN 118734669 IC50 = 1470 nM T05090 CBIY72 118734670 IC50 > 20 ug.mL-1 T05090 C9C7UX 118734705 IC50 = 19680 nM T05090 CI8G4X 118737400 IC50 = 80 nM T05090 C2F8TQ 118737455 IC50 = 532 nM T05090 CZ61KV 118753026 IC50 = 180 nM T05090 CFI23Y 118753027 IC50 = 930 nM T05090 C75LTK 118753189 IC50 = 3300 nM T05090 CB84TO 121278998 IC50 > 50000 nM T05090 C9S5OK 121279020 IC50 > 50000 nM T05090 CIA40K 121472983 IC50 > 10000 nM T05090 CL3M2F 121499152 IC50 = 2280 nM T05090 C93JAV 122177622 IC50 = 149 nM T05090 C5HJ0C 122177623 IC50 > 10000 nM T05090 CW4K2U 122181880 IC50 = 332.1 nM T05090 CK63UH 122181881 IC50 = 319.5 nM T05090 C0H9WU 122181882 IC50 = 2.31 nM T05090 CR3TU6 122181883 IC50 = 332.4 nM T05090 C57VRL 122181884 IC50 = 846.5 nM T05090 C81QDF 122182040 IC50 = 25.01 nM T05090 C2VO8E 122184845 IC50 = 16.65 nM T05090 CGSF80 122184846 IC50 = 21.62 nM T05090 CN4H8Q 122184847 IC50 = 4 nM T05090 CT94PN 122184848 IC50 = 5.42 nM T05090 CI2X8M 122184849 IC50 = 39.67 nM T05090 C5HOK3 122184850 IC50 = 21.2 nM T05090 CZC3Q4 122184851 IC50 = 17.63 nM T05090 CQW6T3 122184852 IC50 = 18.88 nM T05090 CE4M7C 122184853 IC50 = 192 nM T05090 C7MT9U 122184854 IC50 = 40.78 nM T05090 C4AQ5H 122184855 IC50 = 36 nM T05090 C07UQJ 122184856 IC50 = 13.95 nM T05090 CST56N 122184857 IC50 = 92.03 nM T05090 C6K1HJ 122184858 IC50 = 74.42 nM T05090 CG19IO 122185146 IC50 = 69.19 nM T05090 CI4U2H 122185147 IC50 = 107.7 nM T05090 CU47DI 122185148 IC50 = 275.74 nM T05090 C9XMU5 122185149 IC50 = 263.98 nM T05090 C5QCF0 122185150 IC50 = 176.48 nM T05090 CSA1H8 122185151 IC50 = 474.74 nM T05090 CZG70W 122185152 IC50 = 632.54 nM T05090 C28JVO 122192004 IC50 = 9.77 nM T05090 CF2D8U 122192005 IC50 = 3150 nM T05090 C5W8OZ 122376192 IC50 = 2.65 nM T05090 C3V5ND 122550211 IC50 = 439 nM T05090 CW03VD 126582837 IC50 = 65.08 nM T05090 C5UV6J 126582839 IC50 = 26.76 nM T05090 CR9AC4 126582841 IC50 = 113.45 nM T05090 C1HS3A 126582843 IC50 = 20.79 nM T05090 CFI58L 126582907 IC50 = 151.45 nM T05090 CMT02Y 126582908 IC50 > 10000 nM T05090 CE4CI8 127025178 IC50 = 29 nM T05090 CM38EU 127025541 IC50 = 68 nM T05090 C68TYH 127027490 IC50 = 470 nM T05090 CA14VM 127027506 IC50 = 3248.71 nM T05090 CB9PL5 127027507 IC50 > 10000 nM T05090 CBOJ07 127027508 IC50 > 10000 nM T05090 CT18SH 127027509 IC50 = 8861.76 nM T05090 CG7Q3V 127027808 IC50 = 13700 nM T05090 C6JUF9 127027813 IC50 > 30000 nM T05090 CG8NU7 127027995 IC50 = 11 nM T05090 CV07OM 127028943 IC50 = 23 nM T05090 CC6FD8 127034721 IC50 = 960 nM T05090 C4EH3T 127034722 IC50 = 3180 nM T05090 C2YXR7 127034902 IC50 > 5000 nM T05090 C9ZF0D 127035369 IC50 = 1550 nM T05090 C4GI0F 127037614 IC50 = 113 nM T05090 CZ8A1F 127041696 IC50 > 100000 nM T05090 C5D2OJ 127044292 IC50 = 5950 nM T05090 C58KRZ 127044343 IC50 = 19800 nM T05090 C1TYS6 127044344 IC50 = 25900 nM T05090 C3G0SM 127044498 IC50 = 5730 nM T05090 C5CP9M 127045259 IC50 = 6260 nM T05090 CB8HR2 129104138 IC50 > 50000 nM T05090 CCH65A 129104183 IC50 > 50000 nM T05090 CFH8Q4 129104227 IC50 > 50000 nM T05090 C6HM5P 129104349 IC50 > 50000 nM T05090 CZTF90 129104374 IC50 > 50000 nM T05090 CUJ2P5 129104402 IC50 > 50000 nM T05090 CY3I6X 129104426 IC50 > 50000 nM T05090 C2N5JD 132279660 IC50 > 10000 nM T05090 C4L6UZ 132547258 IC50 = 338 nM T05090 CGBR54 132547259 IC50 = 424 nM T05090 CW4MP2 132547260 IC50 = 356 nM T05090 C1YO2Z 132547261 IC50 = 35 nM T05090 CU63DV 132569672 IC50 = 311 nM T05090 C4KE3N 132938351 IC50 = 368 nM T05090 C4UAN3 134129876 IC50 = 333 nM T05090 C25EVA 134129883 IC50 = 59 nM T05090 CWRH43 134129994 IC50 = 191 nM T05090 CK2TM6 134130010 IC50 = 1020 nM T05090 CYW6H1 134130165 IC50 = 33 nM T05090 C8CY7S 134131006 IC50 = 283 nM T05090 CQ7SN8 134131102 IC50 = 256 nM T05090 CYCS54 134131113 IC50 = 722 nM T05090 CQO23I 134131456 IC50 = 181 nM T05090 CHZ8A3 134131564 IC50 = 224 nM T05090 CN9DL4 134132030 IC50 > 10000 nM T05090 CX93QK 134135812 IC50 > 100000 nM T05090 CN8L9J 134136160 IC50 = 530000 nM T05090 C53UTO 134137062 IC50 = 2000 nM T05090 CSX58U 134139437 IC50 > 10000 nM T05090 C75NRQ 134141877 IC50 > 100000 nM T05090 C62SVR 134142119 IC50 > 100000 nM T05090 CLI48U 134143743 IC50 = 5400 nM T05090 CUA26W 134143927 IC50 = 43000 nM T05090 CWRJ15 134147087 IC50 = 20200 nM T05090 C8K0XJ 134147090 IC50 = 280 nM T05090 CQ61SB 134150479 IC50 = 49200 nM T05090 CDX75O 134152551 IC50 = 10700 nM T05090 C2JV5X 134153768 IC50 > 100000 nM T05090 C38DIF 134156853 IC50 = 98000 nM T05090 C4FLQ5 134157355 IC50 > 100000 nM T05090 C1UP3S 134157845 IC50 = 1830 nM T05090 CZV43J 134283792 IC50 = 23000 nM T05090 C62WXO 134283796 IC50 = 37000 nM T05090 CO7K3N 134283799 IC50 = 6000 nM T05090 CBQ17L 134283800 IC50 = 27000 nM T05090 C1Y4TA 134283810 IC50 = 30000 nM T05090 CV2YF7 134283813 IC50 = 42000 nM T05090 C05FVT 134492522 IC50 > 10000 nM T05090 CS1V6A 135367138 IC50 > 50000 nM T05090 CVO59N 135367789 IC50 > 50000 nM T05090 CDY18W 135407493 IC50 > 100000 nM T05090 CW2I4R 135412048 IC50 > 100000 nM T05090 C7U0AV 135412194 IC50 > 100000 nM T05090 CS54TL 135437514 IC50 = 86400 nM T05090 C36MUC 135441620 IC50 > 100000 nM T05090 CRB8M1 135444536 IC50 > 100000 nM T05090 CX5D6J 135446479 IC50 = 15200 nM T05090 C1TOK2 135449197 IC50 > 100000 nM T05090 CW25GL 135462117 IC50 > 100000 nM T05090 CCL28F 135473106 IC50 > 100000 nM T05090 CYA60G 135497781 IC50 > 100000 nM T05090 C01EZF 135567459 IC50 = 68000 nM T05090 CV3QP4 135886613 IC50 = 25.6 nM T05090 C8X5LO 135928012 Ki = 120 nM T05090 CI2YE8 135928628 IC50 > 100000 nM T05090 C50NIS 136025837 IC50 > 100000 nM T05090 C4OS0V 136025842 IC50 > 100000 nM T05090 CX7Z5B 136025843 IC50 > 100000 nM T05090 CB8EM9 136025984 IC50 > 100000 nM T05090 C49MUG 136025986 IC50 > 100000 nM T05090 CH7Y3C 136086920 IC50 > 100000 nM T05090 C3VDL5 136086921 IC50 > 100000 nM T05090 C9GOB5 136086922 IC50 = 40000 nM T05090 CE3ZL7 136086923 IC50 > 100000 nM T05090 CJZ5F3 136086924 IC50 > 100000 nM T05090 CY9U0E 136173089 IC50 = 20 nM T05090 CXHY69 136230092 IC50 = 690 nM T05090 CWK9U7 136230093 IC50 = 410 nM T05090 C7X1UL 136645449 IC50 = 854 nM T05090 CA5OY1 137628667 IC50 = 45 nM T05090 C67EFJ 137628684 IC50 = 1.47 nM T05090 CX0PH5 137628685 IC50 = 654 nM T05090 CG23FD 137631444 IC50 = 10390 nM T05090 C9UQD2 137631509 IC50 > 30000 nM T05090 CP0JL9 137631552 IC50 > 30000 nM T05090 CHL7E8 137631592 IC50 = 8007 nM T05090 CJ9GD5 137631769 IC50 > 30000 nM T05090 CJ7P1U 137631803 IC50 = 227 nM T05090 CQ54WK 137631915 IC50 > 30000 nM T05090 CD1L0I 137632135 IC50 > 30000 nM T05090 C6A4GK 137632422 IC50 > 30000 nM T05090 CQ4BK9 137632561 IC50 > 30000 nM T05090 CVB93K 137632723 IC50 = 1800 nM T05090 C9RWF1 137632979 IC50 > 30000 nM T05090 CI2G7B 137633049 IC50 > 30000 nM T05090 CMU42D 137633092 IC50 > 30000 nM T05090 CY08AM 137633123 IC50 > 30000 nM T05090 C84MIY 137633138 IC50 = 3570 nM T05090 C1HL3I 137633415 IC50 > 30000 nM T05090 CM6V3G 137633491 IC50 = 65.05 nM T05090 C8G4KJ 137634562 IC50 > 30000 nM T05090 CJ76DN 137634596 IC50 > 30000 nM T05090 C7JK8D 137634598 IC50 = 356.9 nM T05090 C7U1CE 137634604 IC50 > 30000 nM T05090 C28CEY 137634881 IC50 = 67.54 nM T05090 C90TSR 137634950 IC50 > 30000 nM T05090 CHA4E3 137635225 IC50 = 1940 nM T05090 CBMN61 137635405 IC50 > 30000 nM T05090 CZ29MT 137635651 IC50 = 5170 nM T05090 COF8J3 137635708 IC50 = 223 nM T05090 C7N5BG 137635855 IC50 > 30000 nM T05090 C2MB4U 137636234 IC50 = 1010 nM T05090 CA2S3J 137636481 IC50 = 220 nM T05090 C5GCO8 137636604 IC50 > 30000 nM T05090 C72SBN 137636632 IC50 > 30000 nM T05090 C9THE6 137636891 IC50 > 30000 nM T05090 CF3E8T 137637310 IC50 > 30000 nM T05090 C0VNM5 137637430 IC50 = 144.07 nM T05090 C6MVX0 137637661 IC50 = 4150 nM T05090 C3H2GO 137637718 IC50 = 750 nM T05090 CSH08B 137637787 IC50 = 2550 nM T05090 CEI0W2 137637915 IC50 = 2900 nM T05090 CZU9E2 137637958 IC50 = 24.71 nM T05090 CMU93I 137637990 IC50 > 30000 nM T05090 C6X0AW 137638091 IC50 = 19.8 nM T05090 CMD89K 137638151 IC50 = 1800 nM T05090 CQ3DR6 137638257 IC50 = 1210 nM T05090 CO9UY1 137638342 IC50 > 30000 nM T05090 C3RC2O 137638626 IC50 > 30000 nM T05090 CEMX30 137638687 IC50 > 30000 nM T05090 CTG6X0 137638748 IC50 > 30000 nM T05090 CZU31H 137638926 IC50 = 850 nM T05090 CQ86FE 137638947 IC50 > 30000 nM T05090 C7IJC2 137639014 IC50 = 430 nM T05090 C2DIM1 137639536 IC50 = 600 nM T05090 CW4DJ8 137639563 IC50 > 30000 nM T05090 CS9A6C 137639566 IC50 > 30000 nM T05090 CMI6Z0 137639764 IC50 = 1030 nM T05090 COV42L 137639829 IC50 > 30000 nM T05090 CL02GC 137640047 IC50 = 1320 nM T05090 C19GDO 137640291 IC50 = 7.1 nM T05090 CGKA54 137640295 IC50 > 30000 nM T05090 C7VIL6 137640304 IC50 = 3100 nM T05090 C0Q3ZW 137640468 IC50 = 12600 nM T05090 C39FQX 137641152 IC50 > 30000 nM T05090 CSA84O 137641263 IC50 = 590 nM T05090 CI4PM3 137641395 IC50 > 30000 nM T05090 C4OEC3 137641520 IC50 = 1600 nM T05090 CS1K3I 137641616 IC50 > 30000 nM T05090 C38HXT 137641735 IC50 = 4940 nM T05090 CV19SL 137642038 IC50 > 30000 nM T05090 CAF1N9 137642211 IC50 = 64.51 nM T05090 C40JZA 137642448 IC50 > 30000 nM T05090 CY02GK 137642671 IC50 > 30000 nM T05090 CF42GI 137643288 IC50 = 152.46 nM T05090 CJOS87 137643760 IC50 = 96 nM T05090 C4V1WC 137643841 IC50 = 830 nM T05090 CB59SN 137643993 IC50 = 147 nM T05090 C7DLO4 137644089 IC50 = 5626 nM T05090 CC38FN 137644424 IC50 > 30000 nM T05090 CVQ4J0 137644605 IC50 > 30000 nM T05090 CX37VS 137644658 IC50 > 30000 nM T05090 CCBN61 137645084 IC50 = 30850 nM T05090 CPL3J1 137645258 IC50 > 30000 nM T05090 C8XAR3 137645372 IC50 > 30000 nM T05090 C05LHW 137645511 IC50 > 30000 nM T05090 CX3E0H 137645675 IC50 = 138 nM T05090 C5REZ8 137645689 IC50 > 20000 nM T05090 CYSU67 137645967 IC50 > 30000 nM T05090 C8HKU4 137646033 IC50 = 98.79 nM T05090 CV7F6C 137646133 IC50 = 180 nM T05090 CMJ7D9 137646202 IC50 > 30000 nM T05090 CN08DL 137646214 IC50 > 30000 nM T05090 CNT3Y7 137647005 IC50 = 196.62 nM T05090 C4I9YE 137647260 IC50 = 5210 nM T05090 CX8C9V 137647325 IC50 > 30000 nM T05090 CHW8X4 137647384 IC50 > 30000 nM T05090 C5AFM1 137647889 IC50 = 50.27 nM T05090 CZ2RN9 137647935 IC50 > 30000 nM T05090 CO7H5A 137648171 IC50 = 151800 nM T05090 C5IK9F 137648357 IC50 = 215.48 nM T05090 C8S2TO 137648573 IC50 = 4310 nM T05090 C0VAB8 137648585 IC50 > 30000 nM T05090 CPK7Y5 137648623 IC50 = 5290 nM T05090 CL0XW1 137648762 IC50 = 660 nM T05090 CR0P6Z 137648837 IC50 = 910 nM T05090 CN3I9X 137648982 IC50 = 90 nM T05090 CG2PL8 137648996 IC50 = 3210 nM T05090 C05DNH 137649390 IC50 > 30000 nM T05090 CO20AE 137649565 IC50 > 30000 nM T05090 C0PGD9 137649617 IC50 = 62540 nM T05090 CH0ES8 137650022 IC50 > 30000 nM T05090 C4MC5X 137650991 IC50 > 30000 nM T05090 C4GNA5 137651338 IC50 > 30000 nM T05090 C8PWX1 137651771 IC50 > 30000 nM T05090 CGE1Z5 137651786 IC50 = 8710 nM T05090 CD89ZR 137651966 IC50 > 30000 nM T05090 C3EQ0D 137651991 IC50 = 33.77 nM T05090 CT05IE 137651994 IC50 = 570 nM T05090 CH3B5G 137652131 IC50 > 30000 nM T05090 C5FHD3 137652442 IC50 = 12500 nM T05090 CMP7G0 137652638 IC50 = 167 nM T05090 C83RBI 137652888 IC50 = 2570 nM T05090 CPI06O 137652951 IC50 = 133.06 nM T05090 C61VOF 137653427 IC50 = 490 nM T05090 C1OAE9 137654162 IC50 = 950 nM T05090 CFQ4T2 137654668 IC50 > 30000 nM T05090 C1SBN5 137654946 IC50 = 6530 nM T05090 CLWF87 137655165 IC50 > 30000 nM T05090 CS50BH 137655597 IC50 > 30000 nM T05090 CIA0V1 137656228 IC50 > 30000 nM T05090 CVG9T3 137656290 IC50 = 19 nM T05090 C0EQI2 137656898 IC50 = 42.9 nM T05090 C76OGQ 137656942 IC50 = 24000 nM T05090 C5BM7T 137657586 IC50 = 110 nM T05090 C97QUM 137657678 IC50 = 243 nM T05090 C21XDS 137657845 IC50 = 5800 nM T05090 CN0C1E 137658519 IC50 > 30000 nM T05090 COC9D2 137658833 IC50 > 30000 nM T05090 CPJL30 137659007 IC50 = 261 nM T05090 CFGW13 137659898 IC50 = 667 nM T05090 C7JGX8 137660397 IC50 = 45.55 nM T05090 C3Q7PX 137660404 IC50 = 1030 nM T05090 C02BSL 137661253 IC50 = 99.87 nM T05090 CQAY45 137662133 IC50 = 4290 nM T05090 CYZ43W 137662281 IC50 = 21.37 nM T05090 CAQ62X 137701235 Ki = 12 nM T05090 CIWG23 138393067 IC50 = 430 nM T05090 C7EM3I 138393071 IC50 = 4150 nM T05090 C4NFS3 138393072 IC50 = 178.3 nM T05090 CIT72O 139302883 IC50 = 3.78 nM T05090 CN1TH8 139302889 IC50 = 189 nM T05090 C0R1MD 139302991 IC50 = 42.51 nM T05090 C3GJQ8 139303021 IC50 = 17.06 nM T05090 CN73DV 139303049 IC50 = 260 nM T05090 CFAU90 139303050 IC50 = 38.41 nM T05090 CKQB30 139303051 IC50 = 13.88 nM T05090 CN2UH1 139303146 IC50 = 3.02 nM T05090 CE81VG 139303149 IC50 = 2.54 nM T05090 C9DJ3B 139303559 IC50 = 11.35 nM T05090 CP73QO 141504704 IC50 = 660 nM T05090 CX0E9B 142505968 IC50 = 10600 nM T05090 CBJC50 142505992 IC50 = 7075 nM T05090 C7N8LV 142506025 IC50 = 1031 nM T05090 CKBF56 142506033 IC50 = 427 nM T05090 CLND62 142506170 IC50 > 100000 nM T05090 CGNQ74 142506189 IC50 = 6699 nM T05090 C1T3IQ 142506210 IC50 = 2400 nM T05090 CXJ0Y4 145949850 IC50 = 32 nM T05090 CKG98W 145953085 IC50 > 30000 nM T05090 CBNG29 145957781 IC50 = 64 nM T05090 CK1XI0 145960971 IC50 > 10000 nM T05090 C3PWD4 145964064 IC50 = 2050 nM T05090 CDY56B 145964885 IC50 = 232 nM T05090 CJAE67 145966594 IC50 = 3910 nM T05090 C19POY 145967140 IC50 = 5090 nM T05090 CSJ81Y 145968726 IC50 = 59.6 nM T05090 CI43DY 145970786 IC50 > 100000 nM T05090 CO51JK 145973368 IC50 = 11.1 nM T05090 C4HTO2 145973543 IC50 = 861 nM T05090 CVM0Z3 145974125 IC50 = 2560 nM T05090 C8YEJ9 145974425 IC50 = 4400 nM T05090 CE8I5V 145975869 IC50 = 323 nM T05090 CMUA94 145976675 IC50 = 891 nM T05090 CN6UO4 145977003 IC50 = 996 nM T05090 CKAQ67 145977127 IC50 = 6050 nM T05090 COR40V 145978805 IC50 = 6620 nM T05090 C9BJW3 145979532 IC50 = 164 nM T05090 CZ7IQ9 145979841 IC50 = 0.41 nM T05090 C0UG8S 145980171 IC50 = 1220 nM T05090 CMB08D 145981960 IC50 = 60.3 nM T05090 C9VDE5 145982499 IC50 = 340 nM T05090 CKYP15 145982514 IC50 = 11780 nM T05090 CX2LY1 145982614 IC50 = 9320 nM T05090 C0SHF9 145982778 IC50 = 12000 nM T05090 CR63YW 145983218 IC50 = 100 nM T05090 C6OL1K 145983267 IC50 = 544 nM T05090 CE38WZ 145983432 IC50 = 1300 nM T05090 CPUJ75 145983482 IC50 = 27310 nM T05090 CWD0A9 145983712 Ki = 0.8 nM T05090 C2I7EQ 145983818 IC50 = 18830 nM T05090 CV8H2B 145983876 IC50 = 25380 nM T05090 C3I6VL 145983950 IC50 = 780 nM T05090 C7FBZ5 145984102 IC50 = 34860 nM T05090 CIWO70 145984314 IC50 = 1810 nM T05090 C9ZKC1 145984665 IC50 = 1890 nM T05090 CSA1K8 145984949 IC50 = 37190 nM T05090 CT50ZG 145985100 IC50 = 1600 nM T05090 CFLH65 145985111 IC50 = 24610 nM T05090 CN6KB9 145985243 IC50 = 160 nM T05090 CK90XR 145985933 IC50 = 100 nM T05090 CBF13W 145985947 IC50 = 5330 nM T05090 C56MWZ 145986208 Ki = 58 nM T05090 CL62QV 145986214 IC50 = 2650 nM T05090 CGN02Q 145986264 IC50 = 990 nM T05090 C51BUM 145986322 IC50 = 0.75 nM T05090 C82CIN 145988785 IC50 = 1500 nM T05090 CHR0U9 145990400 IC50 = 1.3 nM T05090 C68VKC 145993051 IC50 = 1190 nM T05090 C1W6CF 145994016 IC50 = 23000 nM T05090 C0GMR1 146585718 IC50 = 10990 nM T05090 C0YXS8 147254231 IC50 = 3951 nM T05090 CN71OS 149405396 IC50 = 1973 nM T05090 C9FIY4 153534005 IC50 = 75 nM T05090 CB8RS9 155512087 IC50 > 25000 nM T05090 CQ5BL7 155512551 IC50 > 50000 nM T05090 CPF6R7 155512997 IC50 = 213 nM T05090 CE4H7I 155513471 IC50 > 50000 nM T05090 CW3VT9 155514603 IC50 > 50000 nM T05090 CZ84WI 155515284 IC50 > 50000 nM T05090 CUKG21 155515602 IC50 > 50000 nM T05090 CY2DC1 155515836 IC50 = 148 nM T05090 CYJ53T 155515864 IC50 = 20000 nM T05090 CA1J3N 155517086 IC50 = 126 nM T05090 CEH2N5 155518106 IC50 = 235 nM T05090 C41AIO 155518963 IC50 > 1000 nM T05090 CDY5H6 155519645 IC50 = 1440 nM T05090 CAZ3S7 155521187 IC50 = 18000 nM T05090 CZ75FW 155521272 IC50 = 96 nM T05090 CEQ58R 155523224 IC50 = 83 nM T05090 CNW0D1 155524821 IC50 = 76 nM T05090 CN7B1T 155525782 IC50 > 100000 nM T05090 CHR4K5 155528532 IC50 > 100000 nM T05090 C0IC6W 155528706 IC50 = 146 nM T05090 CZ70PO 155529066 IC50 > 50000 nM T05090 C49NGT 155529137 IC50 > 50000 nM T05090 CZMC49 155530597 IC50 = 1.3 nM T05090 COTR30 155530602 IC50 = 708 nM T05090 CN3W5J 155531452 IC50 > 50000 nM T05090 CKV01F 155531688 IC50 = 380 nM T05090 CK2UY4 155531957 IC50 = 50000 nM T05090 CV2C8O 155532194 IC50 = 290 nM T05090 C1F4DU 155533216 IC50 = 680 nM T05090 CIZ46A 155533876 IC50 > 30000 nM T05090 CJH9L4 155535498 IC50 = 503 nM T05090 CAG9P4 155537573 IC50 > 50000 nM T05090 CLD19W 155539311 IC50 = 2060 nM T05090 CU6V4Q 155539319 IC50 > 50000 nM T05090 CP9O4L 155539654 IC50 = 2700 nM T05090 CE6G4A 155539837 IC50 = 16.29 nM T05090 C6U0FM 155540189 IC50 = 26000 nM T05090 CKZ9A5 155543845 IC50 = 276 nM T05090 CP4L1F 155544459 IC50 > 50000 nM T05090 C1VF5A 155544728 IC50 = 213 nM T05090 CXR86J 155545078 IC50 > 50000 nM T05090 CF2O4J 155546325 IC50 > 50000 nM T05090 C0AU1L 155546632 IC50 > 50000 nM T05090 CEF69A 155546817 IC50 = 185 nM T05090 C90FBZ 155549087 IC50 > 50000 nM T05090 CCTU12 155549163 IC50 > 1000 nM T05090 CE0YL6 155549538 IC50 = 30 nM T05090 CFA01C 155549905 IC50 = 148 nM T05090 C4Z5JX 155550827 IC50 = 50000 nM T05090 C05ZVG 155552130 IC50 = 10900 nM T05090 C46WHP 155552329 IC50 > 1000 nM T05090 CS5D0O 155552399 IC50 = 410 nM T05090 CV4Y5B 155552792 IC50 = 160 nM T05090 CGDF76 155554360 IC50 = 24000 nM T05090 CC56ED 155554844 IC50 = 1.7 nM T05090 CXGR50 155555191 IC50 = 60 nM T05090 CFW90N 155555562 IC50 = 4.21 nM T05090 C7QTU1 155555957 IC50 > 50000 nM T05090 CIN57Q 155556138 IC50 = 34 nM T05090 C0IO1Q 155557341 IC50 = 125 nM T05090 CJ9FW6 155557777 IC50 = 374 nM T05090 CJ3MZ1 155558467 IC50 = 372 nM T05090 C8AUB0 155558567 IC50 = 112 nM T05090 C0RZ7V 155558710 IC50 > 1000 nM T05090 C28CVZ 155559279 IC50 = 132 nM T05090 CPD50Q 155559583 IC50 = 1000 nM T05090 CY3XI1 155559600 IC50 > 1000 nM T05090 C4EQ8P 155561585 IC50 = 260 nM T05090 CGL24S 155562249 IC50 > 50000 nM T05090 C4IM1X 155564305 IC50 = 492 nM T05090 CPNA06 155564750 IC50 > 50000 nM T05090 CE0U7K 155564881 IC50 > 1000 nM T05090 CZDC03 155565491 IC50 > 30000 nM T05090 CG65CR 155565674 IC50 = 50000 nM T05090 C3G1JV 155565712 IC50 > 1000 nM T05090 CD05RS 155566122 IC50 = 43000 nM T05090 C4A0RK 155566461 IC50 > 50000 nM T05090 C04CGS 155567444 IC50 > 50000 nM T05090 CS03PJ 155568350 IC50 > 50000 nM T05090 CW5XB4 155569484 IC50 = 60.3 nM T05090 C3BAZ5 24861442 IC50 = 23.9 nM T05090 D00GBB 11449246 Ki = 23 nM T05090 D00HFS 46884057 IC50 = 114 nM T05090 D00HXX 56650312 IC50 = 80 nM T05090 D00SEE 11379392 IC50 = 201 nM T05090 D01FYB 23648267 IC50 > 20000 nM T05090 D01YBR 44591988 IC50 = 4080 nM T05090 D02NWS 279980 Ki = 1650 nM T05090 D03QOD 239512 IC50 > 50000 nM T05090 D04DOL 25032059 IC50 = 7 nM T05090 D04KQF 6675804 Ki = 275 nM T05090 D04UVL 1133083 IC50 = 3640 nM T05090 D05OVV 11993691 IC50 = 350 nM T05090 D07YZZ 5173 Ki = 125 nM T05090 D0B3ZM 11436024 IC50 = 725 nM T05090 D0E0TA 44454650 IC50 > 50000 nM T05090 D0E9DD 16095101 IC50 = 80 nM T05090 D0H7QA 46884056 IC50 = 58 nM T05090 D0K7QR 45269423 IC50 = 18 nM T05090 D0L6YF 46884016 IC50 = 137 nM T05090 D0M9LJ 44454415 IC50 = 11350 nM T05090 D0MD7H 44454143 IC50 = 11000 nM T05090 D0N9AK 44138031 IC50 = 2800 nM T05090 D0Q2CC 46884055 IC50 = 1348 nM T05090 D0Q2GM 44454416 IC50 = 7300 nM T05090 D0Q5DI 71462653 IC50 = 6680 nM T05090 D0Q5MC 24753719 IC50 > 30000 nM T05090 D0R7JA 53344908 IC50 > 43000 nM T05090 D0T0SK 44138032 IC50 = 160 nM T05090 D0T4JQ 264 IC50 = 9000 nM T05090 D0U8FC 759408 IC50 = 2800 nM T05090 D0W1PV 6918328 Ki = 0.26 nM T05090 D0XZ9Q 11149404 IC50 = 110 nM T05090 D0YO6M 785232 IC50 = 1400 nM T05090 D0Z8PX 24757913 IC50 = 245 nM T69563 D07DCG 71657455 IC50 = 7.5 nM T69563 D07GRH 2749 Ki > 50000 nM T69563 D07VYP 118955396 IC50 = 9 nM T69563 D0C6RM 118310260 IC50 < 10 nM T69563 D0K7FT 89683805 IC50 = 4950 nM T69563 D0K9PC 117817422 IC50 = 0.04 nM T69563 D0RZ9V 90415637 IC50 = 18 nM T69563 CK0JI9 1548955 IC50 = 37860 nM T69563 CV7YQ1 2942796 IC50 = 50000 nM T69563 CS9M6R 3047730 Ki > 50000 nM T69563 C4J5IH 3201893 IC50 = 1800 nM T69563 C0E2RO 3202856 IC50 = 390 nM T69563 CASM49 4016538 IC50 = 410 nM T69563 CY0CO2 5495925 Ki = 12000 nM T69563 C0Q3DC 5760176 Ki > 50000 nM T69563 COI9V5 10389037 IC50 = 270 nM T69563 C3V7MQ 13590964 Ki = 120 nM T69563 C2L5SU 13590965 Ki > 50000 nM T69563 CL5JD4 15187131 Ki = 30000 nM T69563 CN17UX 19287893 Ki > 50000 nM T69563 CG0XH9 20158121 Ki = 870 nM T69563 CX61GC 21520193 Ki > 50000 nM T69563 CBM72Z 25220414 Ki = 16700 nM T69563 C5IW0T 25361650 IC50 = 51400 nM T69563 C5TP6Y 44203254 Ki = 17400 nM T69563 CGCJ16 44541205 Ki = 30000 nM T69563 CPR67J 44541206 Ki > 50000 nM T69563 CCE93X 44541208 Ki > 50000 nM T69563 C3V2US 44543378 Ki = 50000 nM T69563 C3L5JM 45270871 IC50 = 1280 nM T69563 C2ILY9 46952127 IC50 = 704 nM T69563 CFG83B 46958630 IC50 = 3320 nM T69563 CKA58Y 46958631 IC50 = 238 nM T69563 CNP8Y2 54618317 IC50 = 190 nM T69563 CPL7Z4 54619107 IC50 = 6300 nM T69563 CFV27I 54619142 IC50 = 1700 nM T69563 C62ZPY 54619179 IC50 = 5300 nM T69563 CGE50Y 54619189 IC50 = 1000 nM T69563 CBP21C 54619212 IC50 = 3900 nM T69563 CQ4CZ7 54619246 IC50 = 600 nM T69563 C59QBG 54619248 EC50 = 300 nM T69563 C45IFU 54619285 IC50 > 20000 nM T69563 CO01JZ 54621040 IC50 = 550 nM T69563 CHY23G 54621327 IC50 = 91 nM T69563 C14LSD 54630941 IC50 = 6400 nM T69563 C48KIZ 54631125 IC50 = 37 nM T69563 CDO2I1 56645146 IC50 = 60 nM T69563 CFC0N1 56645147 IC50 = 60 nM T69563 CV90CE 56645355 IC50 = 80 nM T69563 C3WB8U 56645356 IC50 = 20 nM T69563 C2XV4G 56645357 IC50 = 40 nM T69563 C2AG6K 56646155 IC50 = 140 nM T69563 CPK0W1 56646779 IC50 = 50 nM T69563 C7RNB0 56832448 IC50 = 860 nM T69563 CFU0G9 56832449 IC50 < 100 nM T69563 CFK30C 56844254 IC50 > 57000 nM T69563 C4TE8X 56923423 IC50 = 50 nM T69563 C8LDQ3 66664967 IC50 = 7800 nM T69563 CX7PG5 66665307 IC50 = 900 nM T69563 C2P4KZ 66665324 IC50 = 5640 nM T69563 CS3U4V 68056458 IC50 = 640 nM T69563 CN0X4D 68056459 IC50 = 60 nM T69563 C7UET3 68056593 IC50 = 40 nM T69563 CRN8L7 68056678 IC50 = 420 nM T69563 C7I8YC 68057381 IC50 > 11000 nM T69563 CPBU43 68057382 IC50 = 80 nM T69563 C9OS2V 68057395 IC50 = 240 nM T69563 CEF19C 68057634 IC50 = 60 nM T69563 CNW1D3 71452045 IC50 = 1100 nM T69563 C8U2OI 71452046 IC50 = 1400 nM T69563 CE0WX3 71453859 IC50 = 3600 nM T69563 CR93TM 71453860 IC50 > 100000 nM T69563 C76JOC 71455563 IC50 = 1270 nM T69563 CBR65Z 71457355 IC50 = 1630 nM T69563 C9ZJR0 71457380 IC50 = 450 nM T69563 CV09MQ 71459238 IC50 = 290 nM T69563 CR8ZV7 71460994 IC50 = 140 nM T69563 C16IGX 71461015 IC50 = 2880 nM T69563 C6H5EQ 71461016 IC50 = 53100 nM T69563 CJ6VF9 71462745 IC50 = 570 nM T69563 C60AFH 71462746 IC50 = 190 nM T69563 C0YX6L 71462747 IC50 > 100000 nM T69563 C5K4SM 71533725 IC50 > 57000 nM T69563 C2A5LR 71541908 IC50 = 36 nM T69563 CX6HR5 71542283 IC50 = 39 nM T69563 C24FVX 71542286 IC50 = 14 nM T69563 C3U5RS 71606602 IC50 = 1580 nM T69563 CL4DW0 71816506 Ki = 270 nM T69563 C4H2SI 71816677 Ki = 270 nM T69563 C6JY3X 71816678 Ki = 2400 nM T69563 CO4UL8 73354948 Ki = 120 nM T69563 C8W5JL 73427242 IC50 = 11 nM T69563 C92IJQ 86268389 IC50 = 33 nM T69563 CPJ76F 86269829 IC50 = 4 nM T69563 CCKB17 86269832 IC50 = 30 nM T69563 C5GO6B 86270015 IC50 = 240 nM T69563 CLM23D 86299415 IC50 = 8.45 nM T69563 CEIX57 86299748 IC50 < 100 nM T69563 CO0E9H 86580656 IC50 = 1 nM T69563 CK0DO7 89479018 IC50 = 610 nM T69563 CR2CN8 89489859 IC50 = 94 nM T69563 CBP73I 89489907 IC50 = 820 nM T69563 CK7HO6 89489971 IC50 = 8800 nM T69563 C8J3EW 89684116 IC50 = 78 nM T69563 CR9TK5 89699486 IC50 = 8 nM T69563 C9X0CZ 89699544 IC50 < 100 nM T69563 C43NDF 89699781 IC50 < 100 nM T69563 CC2U5B 89700010 IC50 < 100 nM T69563 CAH2X0 89700075 IC50 < 100 nM T69563 CT1SH4 89700209 IC50 < 100 nM T69563 CFR82W 89711418 IC50 < 100 nM T69563 C21EGI 90422240 IC50 = 10.9 nM T69563 CM51KW 90452084 IC50 = 24 nM T69563 C4CO1H 90454346 IC50 = 22 nM T69563 C2ZPL7 90454349 IC50 = 15 nM T69563 CU12EN 90458225 IC50 < 100 nM T69563 CX7F2H 90466415 IC50 = 4 nM T69563 C5R3IX 91864709 IC50 = 4.6 nM T69563 C1P4KD 97161268 IC50 = 70 nM T69563 CO34YI 101884787 Ki = 150 nM T69563 C7NQB8 101884789 Ki = 340 nM T69563 CL03EK 101884790 Ki = 140 nM T69563 CFO13M 101884791 Ki = 950 nM T69563 CA1V7W 101884792 Ki = 380 nM T69563 C2B8SY 101884793 Ki = 250 nM T69563 CL9ZV3 101884794 Ki = 140 nM T69563 CF3HU5 101884795 Ki = 5600 nM T69563 CP4JS6 101884796 Ki = 4500 nM T69563 CHY62S 117603922 Ki > 50000 nM T69563 CK0NU9 117817076 IC50 = 2 nM T69563 CTA4U5 117817125 IC50 = 4 nM T69563 CM0W3N 117817132 IC50 = 1 nM T69563 CO4E9M 117817141 IC50 = 0.7 nM T69563 CFQ7I2 117817149 IC50 = 7 nM T69563 CI6BN3 117817339 IC50 = 0.25 nM T69563 CGRI81 117817435 IC50 = 0.3 nM T69563 C2R6FU 117817465 IC50 < 50 nM T69563 CXO21M 117817521 IC50 < 50 nM T69563 C3SPF6 117817536 IC50 < 50 nM T69563 CHOA78 117817538 IC50 < 50 nM T69563 C24YMC 118290999 IC50 = 110 nM T69563 CX1E9U 118291067 IC50 > 10000 nM T69563 C1L4YQ 118291499 IC50 = 210 nM T69563 C42UWZ 118291506 IC50 = 1500 nM T69563 CF6ZP1 118291647 IC50 = 1770 nM T69563 CQ78GD 118291683 IC50 = 8000 nM T69563 CJYC54 118310293 IC50 < 10 nM T69563 C89HIP 118310540 IC50 < 10 nM T69563 CK1GM4 118310766 IC50 < 10 nM T69563 CVC47U 118704643 IC50 = 2220 nM T69563 CE1F9G 118716664 IC50 = 7.27 nM T69563 CE8P7S 118716665 IC50 = 194 nM T69563 C4OHN1 118717060 Ki > 50000 nM T69563 CYK47T 118717061 Ki > 50000 nM T69563 CLS3X4 118717062 Ki = 46000 nM T69563 C20HYE 118717063 Ki > 50000 nM T69563 CW86RL 118717064 Ki > 50000 nM T69563 C6INW2 118717065 Ki > 50000 nM T69563 CI0G3J 118717066 Ki > 50000 nM T69563 CB8G2F 118717067 Ki = 10000 nM T69563 CWHK89 118717068 Ki = 27000 nM T69563 CJ9FT2 118717069 Ki = 4500 nM T69563 CCUM32 118717070 Ki = 9500 nM T69563 C0GAK8 118717071 Ki = 16200 nM T69563 CA94XC 118717072 Ki = 13600 nM T69563 CLRI67 118717073 Ki = 5500 nM T69563 CYOP14 118717074 Ki = 560 nM T69563 CNO9A8 118717075 Ki = 490 nM T69563 CKGO91 118717076 Ki = 650 nM T69563 C2CEK1 118717077 Ki = 2200 nM T69563 CY96SX 118717078 Ki = 2200 nM T69563 CMD28R 118717079 Ki = 12500 nM T69563 C1CT8Z 118717080 Ki = 1600 nM T69563 CU65HC 118717081 Ki > 50000 nM T69563 CM9R7E 118717082 Ki = 8500 nM T69563 C63RNW 118717083 Ki = 3200 nM T69563 C1VG8Y 118717084 Ki = 3100 nM T69563 CI5GF3 118717085 Ki = 600 nM T69563 C3YOI1 118717086 Ki = 750 nM T69563 C1AK2U 118717087 Ki = 950 nM T69563 CW36LO 118717088 Ki = 40500 nM T69563 CW4B7P 118717089 Ki = 27500 nM T69563 C14MZQ 118717090 Ki = 22500 nM T69563 CW23YJ 118717091 Ki = 270 nM T69563 CUH05G 118717092 Ki = 300 nM T69563 C6TRH5 118717093 Ki = 3800 nM T69563 CTCY15 118717094 Ki > 50000 nM T69563 CTC48X 118953591 IC50 = 1 nM T69563 C2F0HL 118953746 IC50 = 293 nM T69563 C3FH8U 118953752 IC50 = 9 nM T69563 CGV23R 118953762 IC50 = 43 nM T69563 CAY4W1 118953816 IC50 = 36.5 nM T69563 CIQ51N 118953858 IC50 = 18 nM T69563 C2TCK0 118953878 IC50 = 4 nM T69563 C6TS3A 118953907 IC50 < 10 nM T69563 C0LK2C 118953916 IC50 = 53 nM T69563 COYJ23 118954160 IC50 < 10 nM T69563 CT6ML1 118955389 IC50 = 223 nM T69563 CZ47QL 118955394 IC50 < 2 nM T69563 CS2GZ7 118955397 IC50 = 40.3 nM T69563 C90ETU 118955405 IC50 = 25 nM T69563 C8K1UB 118955416 IC50 = 358 nM T69563 CNWT10 118955424 IC50 = 4 nM T69563 C7NH0V 118955426 IC50 = 8 nM T69563 CV7SM5 118955430 IC50 = 694 nM T69563 CL3E8F 118955433 IC50 < 2 nM T69563 C2HF8P 118955448 IC50 = 160 nM T69563 C64OGA 118955458 IC50 = 64.7 nM T69563 C6L4WS 118955554 IC50 = 127 nM T69563 CJY41H 118955555 IC50 < 10 nM T69563 C0JMT1 118955563 IC50 = 998 nM T69563 CHF8G7 118955568 IC50 = 147 nM T69563 C63JBM 118955570 IC50 = 132 nM T69563 COUV04 118955574 IC50 = 6300 nM T69563 CNS5J9 118955576 IC50 = 1710 nM T69563 C2Z4XH 118955582 IC50 = 54 nM T69563 CV3O8K 118955589 IC50 = 455 nM T69563 C0EMW9 118955592 IC50 = 3710 nM T69563 CVIO61 118955597 IC50 = 32 nM T69563 C8Y2JP 118955601 IC50 = 267 nM T69563 C7ZD3C 118955606 IC50 = 16 nM T69563 C5K3BL 118955607 IC50 < 10 nM T69563 CC27OH 118955611 IC50 = 188 nM T69563 CG61SY 118955613 IC50 = 53 nM T69563 CBL1E3 118955615 IC50 = 481 nM T69563 CQI31L 118955618 IC50 = 56 nM T69563 C2JZ9E 118955625 IC50 = 316 nM T69563 C0I1AG 118955638 IC50 = 303 nM T69563 CWC9E0 118955642 IC50 = 23 nM T69563 CAUM15 118955650 IC50 = 225 nM T69563 C9ZR3Y 118955663 IC50 = 3480 nM T69563 C86JQU 118955667 IC50 = 138 nM T69563 CIDZ73 118955672 IC50 = 13 nM T69563 C4NF7Z 118955679 IC50 = 668 nM T69563 COU0K5 118955687 IC50 = 69 nM T69563 C2N8CB 118955691 IC50 = 913 nM T69563 C1W6RT 118955698 IC50 = 464 nM T69563 C5RCP1 118955701 IC50 = 77 nM T69563 COS41X 118955712 IC50 = 3110 nM T69563 C1XWG9 118955715 IC50 = 140 nM T69563 C5XVE9 118955721 IC50 = 76 nM T69563 CT24YZ 118955730 IC50 = 995 nM T69563 C5XLV0 118955734 IC50 = 382 nM T69563 CW81VD 118955741 IC50 = 231 nM T69563 CR74DW 118955742 IC50 = 9670 nM T69563 CLA3U0 118955743 IC50 = 487 nM T69563 CK2U0H 118955980 IC50 = 100.2 nM T69563 C15GHE 118956024 IC50 = 295 nM T69563 CH39KW 118956036 IC50 = 19300 nM T69563 CNL73Q 118956065 IC50 = 147 nM T69563 CQ5A6C 118956067 IC50 = 92 nM T69563 CW5A8Z 118956116 IC50 = 25000 nM T69563 CTQO83 118956124 IC50 = 344 nM T69563 CC60WG 118956129 IC50 = 365 nM T69563 C5T8NV 118956132 IC50 = 72 nM T69563 CYN69B 118956147 IC50 = 17 nM T69563 CT6X2G 118956170 IC50 = 1260 nM T69563 CK26OG 118956187 IC50 = 185.1 nM T69563 C5YNM0 118956202 IC50 = 5200 nM T69563 CKP1O6 118956227 IC50 = 20 nM T69563 CT58YU 121225870 IC50 > 57000 nM T69563 C2OV0L 121457603 IC50 > 57000 nM T69563 CB80PQ 121457701 IC50 > 57000 nM T69563 CLKW12 121457751 IC50 = 47400 nM T69563 C6ZTQ1 121457762 IC50 > 57000 nM T69563 CT82GB 121461607 IC50 = 33500 nM T69563 C1LDQ5 121461684 IC50 > 57000 nM T69563 CW62PD 121461708 IC50 > 57000 nM T69563 CEY1H9 121461710 IC50 = 33500 nM T69563 C42KHQ 121461721 IC50 > 57000 nM T69563 C2WU8I 121461723 IC50 > 57000 nM T69563 C1OZ2D 121461729 IC50 = 47400 nM T69563 COED87 121461743 IC50 > 57000 nM T69563 CT7PM0 121461757 IC50 > 57000 nM T69563 CV3L8S 121461774 IC50 > 57000 nM T69563 CMS1Q6 121461818 IC50 > 57000 nM T69563 CJG3D2 121461820 IC50 = 47400 nM T69563 CW8R2L 121461821 IC50 = 26600 nM T69563 CAM9R6 122186444 Ki > 50000 nM T69563 C2VYR3 122186445 Ki > 50000 nM T69563 CKX7M4 122186446 Ki = 13400 nM T69563 CC0P2W 122186447 Ki > 50000 nM T69563 CX9I1G 122186448 Ki > 50000 nM T69563 C0KT5U 122186449 Ki = 4800 nM T69563 CKP7G9 122186450 Ki = 9200 nM T69563 COG86J 122186451 Ki = 3600 nM T69563 CUC87V 122186452 Ki = 25000 nM T69563 CU5K8E 122186453 Ki = 750 nM T69563 C06PJL 122186454 Ki = 7800 nM T69563 C7QU8K 122186455 Ki = 420 nM T69563 CV3O7K 122186456 Ki > 50000 nM T69563 C1YDE3 122186457 Ki > 50000 nM T69563 C37CMN 122186458 Ki = 470 nM T69563 CGND61 122186459 Ki = 4600 nM T69563 CB81IV 122186460 Ki = 4300 nM T69563 C4UT5O 122186461 Ki = 5900 nM T69563 CJD79O 122186462 Ki = 25300 nM T69563 C2LNI6 122186463 Ki > 50000 nM T69563 C4C5QG 122186464 Ki = 34200 nM T69563 COT4C2 122186465 Ki = 11300 nM T69563 C80UNC 122186466 Ki = 2600 nM T69563 CPF8Q6 122186467 Ki = 9200 nM T69563 CGH60B 122186468 Ki > 50000 nM T69563 C0HB1P 122186469 Ki = 5600 nM T69563 CUO13Z 122186470 Ki = 3200 nM T69563 CAW9R2 122186471 Ki > 50000 nM T69563 CD26IH 122186472 Ki = 3100 nM T69563 CDC3Y1 122186473 Ki > 50000 nM T69563 C5AZ1C 122186474 Ki > 50000 nM T69563 CUJT30 122186477 Ki = 16500 nM T69563 C1AU6W 126540084 IC50 < 100 nM T69563 C3BR0C 126540358 IC50 < 100 nM T69563 C6O4DK 126540561 IC50 < 100 nM T69563 CA91IL 129080665 IC50 < 10 nM T69563 CEG3X2 129080727 IC50 < 10 nM T69563 CP5K7B 129080745 IC50 < 10 nM T69563 C5DOP3 129102401 IC50 = 3.5 nM T69563 CSH3V4 130356715 IC50 = 2 nM T69563 CY65ND 130418263 IC50 > 10000 nM T69563 C45PYN 130469646 IC50 < 100 nM T69563 CL01PO 130469826 IC50 < 100 nM T69563 CCMJ13 131955127 IC50 = 29800 nM T69563 C4BRM1 132212317 IC50 = 8.89 nM T69563 C1JK0W 132219367 IC50 < 100 nM T69563 CM81VB 132219371 IC50 < 100 nM T69563 CPM48R 132219770 IC50 < 100 nM T69563 CK1DI3 134132786 IC50 = 60 nM T69563 C9JG7W 134135029 IC50 = 260 nM T69563 CML85T 134136251 IC50 = 320 nM T69563 C39BMU 134136448 IC50 = 80 nM T69563 CIQ6Z8 134137347 IC50 = 19000 nM T69563 CFMG90 134140713 IC50 = 1000 nM T69563 CYF9N7 134141391 IC50 = 140 nM T69563 CH6J4X 134141647 IC50 = 32 nM T69563 CUF9M5 134141685 IC50 = 1600 nM T69563 CATD87 134142306 IC50 = 7900 nM T69563 CPCG95 134143587 IC50 = 140 nM T69563 C13YMT 134144334 IC50 = 1400 nM T69563 CO4D1Q 134145417 IC50 = 3100 nM T69563 CR84NZ 134145925 IC50 = 90 nM T69563 CTV9B8 134146140 IC50 = 160 nM T69563 CG7V6W 134146450 IC50 = 7400 nM T69563 CATO08 134147599 IC50 = 96 nM T69563 CXH8W3 134149147 IC50 = 360 nM T69563 CF9NA0 134149890 IC50 > 20000 nM T69563 C5ZLU2 134151046 IC50 = 75 nM T69563 CN6S0J 134151358 IC50 = 11000 nM T69563 CO74YZ 134152117 IC50 = 7700 nM T69563 CD5O3M 134152198 IC50 = 440 nM T69563 C81ESC 134153452 IC50 = 1600 nM T69563 COLF87 134153477 IC50 = 5700 nM T69563 C07YDQ 134153794 IC50 = 9100 nM T69563 CGC6P4 134153864 IC50 = 160 nM T69563 CIHC43 134154520 IC50 = 91 nM T69563 CAC65I 134155569 IC50 = 56 nM T69563 C5U2VM 134156397 IC50 = 28 nM T69563 CL1H7K 134464493 IC50 < 100 nM T69563 CW73JK 134693801 IC50 = 120 nM T69563 CKMU89 134693804 IC50 = 41 nM T69563 CL51MJ 136110950 Ki > 50000 nM T69563 CZF18P 136110951 Ki > 50000 nM T69563 CW3T4O 137333448 IC50 = 21 nM T69563 CAH41F 137440052 IC50 < 100 nM T69563 CQ19ZS 137496890 IC50 < 20 nM T69563 C3XTO9 137548127 IC50 < 300 nM T69563 CG5HS1 138753630 IC50 > 10000 nM T69563 CE0UK8 138976844 IC50 = 8.9 nM T69563 CHA68B 139373943 IC50 < 300 nM T69563 CLC12T 140267775 IC50 = 11 nM T69563 C0NQO6 140267826 IC50 = 1 nM T69563 CQYI50 140267835 IC50 = 3 nM T69563 CW1O0F 140267861 IC50 = 1 nM T69563 CC26QP 141451166 IC50 = 140 nM T69563 CR82BZ 141451167 IC50 = 950 nM T69563 C8TZ6R 141451170 IC50 = 230 nM T69563 C0Q2WJ 141451172 IC50 = 90 nM T69563 CZP73S 141451178 IC50 = 4420 nM T69563 C1FJ8M 141451182 IC50 = 50 nM T69563 C5N3VP 141451185 IC50 = 930 nM T69563 CG93ER 141451187 IC50 = 13620 nM T69563 C5HZB7 141451189 IC50 = 810 nM T69563 CB8W0Q 141492780 IC50 < 100 nM T69563 CJ6S4B 141503237 IC50 < 10 nM T69563 CM8ZT0 141503247 IC50 = 49 nM T69563 CUT16P 141503256 IC50 > 1000 nM T69563 CMB72E 141503257 IC50 = 5.6 nM T69563 CF35VQ 141503261 IC50 = 14 nM T69563 CW9D8I 142547299 IC50 < 20 nM T69563 C6V3PC 145426709 IC50 = 338 nM T69563 C3FJ1U 145426710 IC50 = 138 nM T69563 CPWT56 145426714 IC50 = 5 nM T69563 CT9J1D 145426720 IC50 = 95 nM T69563 C3UDY4 145426748 IC50 = 180 nM T69563 CU0Q3N 145426790 IC50 = 9 nM T69563 CW10RV 145426839 IC50 = 635 nM T69563 CXWN78 145426877 IC50 = 255 nM T69563 CISY09 145426959 IC50 = 266 nM T69563 C8TSE3 145426981 IC50 = 25 nM T69563 CVC37N 145426988 IC50 = 148 nM T69563 CPL8E6 145427034 IC50 = 21 nM T69563 CV63QK 145427036 IC50 = 186 nM T69563 C6BZA7 145427057 IC50 = 172 nM T69563 C8X0YZ 145427073 IC50 = 51 nM T69563 CP96LO 145721285 IC50 = 17310 nM T69563 CG58CF 145721286 IC50 > 50000 nM T69563 CRMU49 145721287 IC50 > 50000 nM T69563 C2IFB6 145721288 IC50 > 50000 nM T69563 CR53AV 145721289 IC50 > 50000 nM T69563 C2A4EJ 145721290 IC50 > 50000 nM T69563 C6X0NF 145950670 IC50 < 2 nM T69563 CLTN42 145951582 IC50 = 14 nM T69563 CBZ59V 145951646 IC50 = 47 nM T69563 CF5X9J 145954559 IC50 = 73 nM T69563 CUR5N4 145954702 IC50 = 145 nM T69563 CXR2W3 145955203 IC50 = 15 nM T69563 C8OM3X 145956839 IC50 = 116 nM T69563 C6HQJ5 145961862 IC50 = 42 nM T69563 C54CSY 145961866 IC50 = 41 nM T69563 C3M9NW 145963523 IC50 = 28 nM T69563 C7GC3U 145963920 IC50 > 10000 nM T69563 CM0T9L 145964379 IC50 = 560 nM T69563 CCM4K8 145965456 IC50 > 10000 nM T69563 CDM3X9 145965619 IC50 = 15 nM T69563 C7FR6H 145966084 IC50 > 10000 nM T69563 C6AM2R 145966168 IC50 = 27 nM T69563 C2FH9U 145966444 IC50 > 1000 nM T69563 CY7BQ5 145966713 IC50 = 15 nM T69563 C1T0UW 145971297 IC50 = 84 nM T69563 C8QCN3 145971400 IC50 = 13 nM T69563 CH50IP 145971583 IC50 = 21 nM T69563 C8P6QC 145971862 IC50 = 2965 nM T69563 C4L0VB 145972381 IC50 = 47 nM T69563 CSK1D4 145972835 IC50 = 42 nM T69563 CRH47A 145973499 IC50 = 260 nM T69563 C75YBO 145974168 IC50 = 275 nM T69563 C8WS0M 145974512 IC50 = 50 nM T69563 CC92FX 145975511 IC50 = 40 nM T69563 C7HVI9 145975779 IC50 = 270 nM T69563 C0VZ4H 145975944 IC50 = 2605 nM T69563 CS6X3V 145976283 IC50 = 108 nM T69563 CCY80A 145976820 IC50 = 22 nM T69563 CCY85M 145978022 IC50 = 128 nM T69563 C73HRS 145978840 IC50 = 19 nM T69563 C5J8NI 145980147 IC50 > 50000 nM T69563 CVJD53 145980478 IC50 = 34 nM T69563 CG0DS6 145980657 IC50 = 46 nM T69563 C1AOH7 145980705 IC50 = 32000 nM T69563 CVZS80 145981016 IC50 > 50000 nM T69563 CX35RT 145981660 IC50 > 50000 nM T69563 CBU6X1 145981803 IC50 > 50000 nM T69563 CAF30W 145981971 IC50 = 40 nM T69563 CREN84 145982246 IC50 = 8 nM T69563 CQS73W 145983417 IC50 = 13310 nM T69563 CBZ54K 145987434 IC50 = 230 nM T69563 CB1A0K 145987773 IC50 > 50000 nM T69563 CX6G9K 145987904 IC50 > 50000 nM T69563 CG39VW 145988250 IC50 > 50000 nM T69563 C3M8WP 145989869 IC50 = 297 nM T69563 C53EQF 145990414 IC50 = 23100 nM T69563 CTDA70 145992655 IC50 > 50000 nM T69563 CSKG09 145993293 IC50 = 45 nM T69563 CIZ83X 145993302 IC50 = 44 nM T69563 C6PR9F 145994156 IC50 > 50000 nM T69563 CJ12IY 146774513 IC50 = 18.8 nM T69563 C8FJ3A 148054621 IC50 = 16.3 nM T69563 CHK41W 149984817 IC50 = 61.9 nM T69563 CUY4O2 151050871 IC50 = 2.3 nM T69563 CU6FL5 151060963 IC50 = 24.1 nM T69563 CRN0K3 151095070 IC50 = 4 nM T69563 C1UW8G 151614103 IC50 = 9.7 nM T69563 C1ATK8 151745584 IC50 = 17.3 nM T69563 CP7B3F 152297087 IC50 = 24.8 nM T69563 CLC50D 152682805 IC50 = 8 nM T69563 CWA1K4 153354193 IC50 = 14.2 nM T69563 C7Z1RB 153354194 IC50 = 128.5 nM T69563 CXC8G3 153354195 IC50 = 43.5 nM T69563 CQ7R2X 153354196 IC50 = 5858 nM T69563 C3GLD4 153354197 IC50 = 9.4 nM T69563 C1CQ5W 153354198 IC50 = 119.1 nM T69563 C1KR3B 153354200 IC50 = 15 nM T69563 CJ2NI6 153354201 IC50 = 23.8 nM T69563 CS7OY3 153354202 IC50 = 1 nM T69563 CKD1H3 153354205 IC50 = 2.1 nM T69563 CC0T9V 153354208 IC50 = 2.12 nM T69563 CU3OF1 154709431 IC50 = 11660 nM T69563 CWKY46 154709433 IC50 = 13310 nM T69563 CB8F9R 155511968 IC50 = 90 nM T69563 CVF25J 155513757 IC50 = 2 nM T69563 C1YT5V 155514864 IC50 = 12 nM T69563 CLH3W0 155515484 IC50 = 112 nM T69563 CH24MR 155515991 IC50 = 1980 nM T69563 CDK81A 155516285 IC50 > 10000 nM T69563 CLJ5H1 155516944 IC50 = 21 nM T69563 CF60TJ 155517478 IC50 = 42 nM T69563 CT2Z8D 155518356 IC50 = 10 nM T69563 C53FQM 155518762 IC50 > 50000 nM T69563 CO4I8L 155519528 IC50 > 50000 nM T69563 C48QWJ 155519945 IC50 < 100 nM T69563 CT94CM 155520089 IC50 > 100000 nM T69563 C06QWY 155520182 IC50 > 50000 nM T69563 C4YO6W 155520615 IC50 = 28 nM T69563 C8A9HN 155520995 IC50 = 12790 nM T69563 CH7ZC1 155521584 IC50 < 100 nM T69563 C29SCL 155522425 IC50 = 3000 nM T69563 C4BK7X 155523227 IC50 = 11860 nM T69563 C1Y2MB 155523310 IC50 = 5000 nM T69563 COZ4K9 155524250 IC50 = 1400 nM T69563 CZ0CD8 155524347 IC50 = 8500 nM T69563 CC5W9E 155524570 IC50 > 200000 nM T69563 CZC8X9 155524600 IC50 = 32 nM T69563 C3VBJ1 155525283 IC50 > 50000 nM T69563 C8QA0B 155525540 IC50 = 290 nM T69563 CAD91T 155526125 IC50 = 81.5 nM T69563 C3LK2Q 155527455 IC50 = 50 nM T69563 CBR52U 155527494 IC50 > 100000 nM T69563 CO9UA0 155528439 IC50 = 38 nM T69563 C4H6ET 155529102 IC50 = 26.6 nM T69563 CPWO50 155529490 IC50 = 1450 nM T69563 CH3SC8 155531040 IC50 = 18000 nM T69563 C4XLB5 155531880 IC50 = 7910 nM T69563 CC2V9G 155532071 IC50 = 21 nM T69563 C30LMB 155532656 IC50 = 190 nM T69563 C4YFQ9 155533059 IC50 = 65 nM T69563 CAP54S 155533635 IC50 = 100 nM T69563 C8HL6B 155533681 IC50 = 2.2 nM T69563 CP9WL2 155533930 IC50 = 28 nM T69563 CJ2GF8 155534982 IC50 = 3050 nM T69563 CVE7U9 155534983 IC50 = 54 nM T69563 CL02MX 155536249 IC50 = 1480 nM T69563 C5LN0G 155536622 IC50 = 55500 nM T69563 CPS53T 155536735 IC50 < 10 nM T69563 C0BQ5V 155537997 IC50 = 18 nM T69563 CV1AE4 155538180 IC50 = 60 nM T69563 CS3X5Z 155540428 IC50 = 831 nM T69563 COAE19 155540545 IC50 = 55 nM T69563 CK4S2B 155540581 IC50 = 250 nM T69563 CQD6E7 155543356 IC50 = 266 nM T69563 C71CUQ 155544473 IC50 < 100 nM T69563 C1GJ2X 155546130 IC50 > 100000 nM T69563 CU1ST0 155547033 IC50 = 3720 nM T69563 CN46TF 155547202 IC50 = 25000 nM T69563 C5GK8W 155547940 IC50 > 25000 nM T69563 CIDO95 155548480 IC50 > 50000 nM T69563 CP27OJ 155548685 IC50 > 25000 nM T69563 C2S3OI 155548929 IC50 < 100 nM T69563 C9Z1RB 155549401 IC50 = 410 nM T69563 CG73WV 155549530 IC50 = 1540 nM T69563 C6UG0I 155549731 IC50 > 50000 nM T69563 CZ9AV3 155550739 IC50 < 100 nM T69563 C48VPJ 155553143 IC50 = 18 nM T69563 CJX6U0 155553326 IC50 > 100000 nM T69563 C18PRB 155553562 IC50 = 44.5 nM T69563 C7KJ4E 155553804 IC50 = 721 nM T69563 C4HT0M 155553871 IC50 = 39600 nM T69563 C7S1AK 155556534 IC50 = 26 nM T69563 C42KSY 155556957 IC50 = 4800 nM T69563 CD7IO6 155556974 IC50 = 82 nM T69563 C5KP4J 155557173 IC50 = 60 nM T69563 CRO21A 155557415 IC50 > 50000 nM T69563 C8AFH6 155557755 IC50 = 152 nM T69563 CV4H2Z 155559814 IC50 > 10000 nM T69563 CU8W4A 155560336 IC50 = 930 nM T69563 CKPE98 155561191 IC50 < 300 nM T69563 C27QFZ 155562355 IC50 > 10000 nM T69563 CHC0E2 155562949 IC50 = 800 nM T69563 C4FZ6B 155563652 IC50 = 50000 nM T69563 C26LSZ 155563728 IC50 = 393.9 nM T69563 CR3WQ5 155565507 IC50 = 43580 nM T69563 CDYB38 155565613 IC50 = 45300 nM T69563 CS01QM 155565995 IC50 > 50000 nM T69563 C5VZN7 155567367 IC50 = 220 nM T69563 D05IWY 5464078 Ki = 3170 nM T69563 D06PRC 5281650 Ki = 2850 nM T70539 D0A3CL 49801838 IC50 > 40000 nM T70539 CYIT28 9806086 IC50 = 10000 nM T70539 C5RIY7 9824428 IC50 > 100000 nM T70539 CTUO16 9955811 IC50 = 6310 nM T70539 CQL12P 10004545 IC50 > 10000 nM T70539 C6OI1A 10005009 IC50 = 6.8 nM T70539 CI8FM2 10025150 IC50 = 100 nM T70539 CS14OM 10027853 IC50 = 4.7 nM T70539 C9QZ0I 10046992 IC50 = 4 nM T70539 CR1ME4 10090198 IC50 = 100 nM T70539 CU7TP2 10091316 IC50 = 10 nM T70539 CG7Z9I 10128764 Ki > 3000 nM T70539 CEO59I 10129026 Ki > 3000 nM T70539 CW5O4B 10129036 Ki > 3000 nM T70539 C3FS7G 10129058 Ki > 3000 nM T70539 CJ05QL 10129135 Ki > 3000 nM T70539 CX9EI2 10143421 Ki > 3000 nM T70539 CZ95DQ 10143980 Ki > 3000 nM T70539 C2X9YI 10152629 Ki > 3000 nM T70539 C9VP5L 10152726 Ki > 3000 nM T70539 CVGB64 10152879 Ki > 3000 nM T70539 CZQ69G 10165656 Ki > 3000 nM T70539 C9EJT4 10166088 Ki > 3000 nM T70539 CC2F7Z 10173787 IC50 = 960 nM T70539 CM9KF2 10174522 Ki > 3000 nM T70539 CH25WF 10174984 Ki > 3000 nM T70539 C47RGT 10186370 Ki > 3000 nM T70539 C80YEW 10188732 Ki > 3000 nM T70539 CGJ7D9 10195667 Ki > 3000 nM T70539 C9OB3S 10196098 Ki > 3000 nM T70539 C2K1LR 10196214 Ki > 3000 nM T70539 CBX4C2 10196316 Ki > 3000 nM T70539 CD9N3H 10196460 Ki > 3000 nM T70539 CYT8S5 10196576 Ki > 3000 nM T70539 C5EGZ8 10196608 Ki > 3000 nM T70539 C0OB2A 10196742 Ki > 3000 nM T70539 CIC0H8 10218194 Ki > 3000 nM T70539 CH7BP9 10218547 Ki > 3000 nM T70539 CX7KR8 10218604 Ki > 3000 nM T70539 CEO3C0 10230947 Ki > 3000 nM T70539 C2AV9K 10239389 Ki > 3000 nM T70539 CWTM13 10239448 Ki > 3000 nM T70539 CY3B9V 10239505 Ki > 3000 nM T70539 C9ZR5W 10239639 Ki > 3000 nM T70539 C8R7NE 10239929 Ki > 3000 nM T70539 C2JY5L 10239930 Ki > 3000 nM T70539 CNY7O0 10280331 Ki > 3000 nM T70539 C7GFV9 10281308 Ki > 3000 nM T70539 CQAM65 10289494 Ki > 3000 nM T70539 CP4MX9 10303281 Ki > 3000 nM T70539 C5NVX2 10310772 Ki > 3000 nM T70539 C8X2OD 10311260 Ki > 3000 nM T70539 CS5YX7 10311798 Ki > 3000 nM T70539 CHR1A3 10312086 Ki > 3000 nM T70539 CCRI74 10312244 Ki > 3000 nM T70539 CMC1G5 10319824 IC50 > 100000 nM T70539 CVO3N7 10344176 IC50 > 10 nM T70539 CL83KQ 10388797 IC50 = 3.7 nM T70539 C6UO4Y 10410064 IC50 = 0.1 nM T70539 C6T7WB 10434776 IC50 > 100000 nM T70539 CFV7D4 10436090 IC50 = 10000 nM T70539 CGS89V 10455647 IC50 = 4 nM T70539 C07KPU 10456755 IC50 > 10 nM T70539 C38VGA 10457264 IC50 = 1 nM T70539 CUD3I6 11156790 Ki > 3000 nM T70539 C19UHW 11168186 Ki > 3000 nM T70539 CPS26T 11201645 IC50 = 6.4 nM T70539 CK9E2Y 11317465 Ki > 3000 nM T70539 CO7CX6 11318577 Ki > 3000 nM T70539 CCU9P8 11318709 Ki > 3000 nM T70539 CB51KQ 11433168 Ki > 3000 nM T70539 C6L8DU 11495754 IC50 > 10 nM T70539 C9YME5 11496313 IC50 > 10 nM T70539 C2B6YR 11512135 IC50 = 4.5 nM T70539 CQ08DH 11539632 IC50 = 8.7 nM T70539 CX6IL5 11548234 IC50 = 6.3 nM T70539 C59SVL 11563383 IC50 > 10 nM T70539 CPA3J7 11583744 IC50 = 7.1 nM T70539 CKI9D5 11599973 IC50 = 4600 nM T70539 CDA48G 11613696 Ki > 3000 nM T70539 C5A4YW 11648240 IC50 = 8.4 nM T70539 CP09GF 11655872 IC50 > 10 nM T70539 CFB78R 11752339 Ki > 3000 nM T70539 CX20YM 11785261 Ki > 3000 nM T70539 CJZ1S6 11785262 Ki > 3000 nM T70539 CL50KS 15983730 Ki > 10000 nM T70539 CB0JD2 16037921 Ki > 3000 nM T70539 C7K5AW 16721015 IC50 > 10000 nM T70539 CBR6Q7 20608969 Ki > 3000 nM T70539 COF9E8 20608974 Ki > 3000 nM T70539 CWSB30 20608975 Ki > 3000 nM T70539 C7PL9M 20608976 Ki > 3000 nM T70539 CG9R3I 20608977 Ki > 3000 nM T70539 C9U6JQ 20608981 Ki > 3000 nM T70539 CC1RB9 20608989 Ki > 3000 nM T70539 C2H1YF 20608991 Ki > 3000 nM T70539 C8Q0XO 20608992 Ki > 3000 nM T70539 C8CUT0 20608996 Ki > 3000 nM T70539 CVGY56 20609011 Ki > 3000 nM T70539 C7N6XY 20609018 Ki > 3000 nM T70539 C78UWI 20609028 Ki > 3000 nM T70539 CKHG76 23572819 IC50 = 30 nM T70539 C2DIJ7 23573799 Ki > 3000 nM T70539 CRCF01 30979231 IC50 = 1000 nM T70539 CMY45F 44188279 Ki > 9700 nM T70539 C76ONX 44219756 IC50 > 1000 nM T70539 C1RD0C 44394909 IC50 > 100000 nM T70539 C0KLA9 44394921 IC50 > 100000 nM T70539 CI7RP8 44394922 IC50 > 100000 nM T70539 C2KM0Q 44394959 IC50 > 100000 nM T70539 CUQ04R 44395076 IC50 = 2880 nM T70539 C4HR6C 44399507 Ki > 3000 nM T70539 CH39TA 44399610 Ki > 3000 nM T70539 CLGA83 44403765 IC50 = 6.8 nM T70539 CD3FE4 44405399 Ki > 3000 nM T70539 CW5KU8 44405417 Ki > 3000 nM T70539 CVP74K 44405418 Ki > 3000 nM T70539 C0N4IL 44405421 Ki > 3000 nM T70539 C79OPX 44405435 Ki > 3000 nM T70539 CDJF17 44405436 Ki > 3000 nM T70539 CT42XM 44405437 Ki > 3000 nM T70539 CF57KL 44405439 Ki > 3000 nM T70539 C37XOM 44405444 Ki > 3000 nM T70539 CW80JL 44405461 Ki > 3000 nM T70539 CN4KP9 44405501 Ki > 3000 nM T70539 CFSD50 44412624 Ki > 3000 nM T70539 C1CPT2 44412682 Ki > 3000 nM T70539 CG6J5R 44412683 Ki > 3000 nM T70539 CQ7P1N 44412686 Ki > 3000 nM T70539 CVJF97 44412837 Ki > 3000 nM T70539 CRPQ04 44412852 Ki > 3000 nM T70539 CV1ZX4 44412960 Ki > 3000 nM T70539 CAQ2D8 45487653 IC50 > 10 nM T70539 CN58HC 57391501 IC50 = 10 nM T70539 C0J6GT 57391502 IC50 = 678 nM T70539 C1W8ZE 57394991 IC50 = 250 nM T70539 CMNZ07 57394992 IC50 = 1 nM T70539 CAID96 57396733 IC50 = 15000 nM T70539 C8AOK6 57396734 IC50 = 200 nM T70539 CO0C6Y 57396735 IC50 = 10 nM T70539 CVN98L 57400176 IC50 = 300 nM T70539 CFXM54 57400177 IC50 = 200 nM T70539 CS05AF 57400178 IC50 = 80 nM T70539 C0SY9X 57400179 IC50 = 150 nM T70539 CRHS14 57400180 IC50 = 8 nM T70539 C98HEK 57401966 IC50 = 60000 nM T70539 CBEW17 57401967 IC50 = 100 nM T70539 C1E2LP 57401968 IC50 = 0.1 nM T70539 CS63IW 57401969 IC50 = 13 nM T70539 C9DF5Y 57403720 IC50 = 10000 nM T70539 C9PN3B 57403721 IC50 = 60000 nM T70539 CXZQ20 57403722 IC50 = 70 nM T70539 CH5EV8 57403723 IC50 = 250 nM T70539 D01NOZ 16665072 IC50 > 30000 nM T75888 D00SBN 4746 IC50 > 100000 nM T75888 D0L5WM 2157 IC50 > 100000 nM T75888 D0Q4YI 21109 IC50 > 100000 nM T75888 D01FCK 9843897 IC50 = 5400 nM T75888 D0P9JW 121830 IC50 > 100000 nM T75888 CSI0D4 355 IC50 = 11000 nM T75888 COK56H 36143 IC50 > 100000 nM T75888 CAUV41 11979264 IC50 = 6400 nM T75888 CY7XM3 13671155 IC50 = 21700 nM T75888 CFD2E4 15234003 IC50 = 160 nM T75888 CZ9JM6 15984085 IC50 > 100000 nM T75888 C7E2FM 16718554 IC50 = 3400 nM T75888 C7ZY1S 16736346 IC50 > 100000 nM T75888 C2WJQ5 23695524 IC50 > 50000 nM T75888 CMFN27 23729161 IC50 = 85300 nM T75888 CMW4E2 24825719 IC50 = 3500 nM T75888 C9KS1T 25095157 IC50 > 100000 nM T75888 CLS8H0 66857424 IC50 > 100000 nM T75888 CQR5T1 71457921 IC50 = 360 nM T15636 CV63UL 67240318 IC50 > 10000 nM T15636 C2MD1Q 155513187 IC50 > 10000 nM T15636 C41NLP 155544908 IC50 = 120 nM T15636 D0VC0I 5169 IC50 = 47200 nM T13453 CZ63PR 16133811 IC50 = 0.8 nM T13453 CP42JF 25180487 Ki = 22 nM T13453 C5VA6W 25180488 Ki = 108 nM T13453 CZ51CD 25180490 Ki = 65.5 nM T13453 C1IU8X 25180491 Ki = 15 nM T13453 C2WMX8 25180492 Ki = 75 nM T13453 CZ1N7I 25180493 Ki = 24 nM T13453 C3G8OJ 25180494 Ki = 28 nM T13453 CHRV59 25180496 Ki = 51 nM T13453 CVN29B 25180497 Ki = 214.5 nM T13453 C62QZX 25180498 Ki = 1323.5 nM T13453 C4DL5C 44469677 IC50 > 10000 nM T13453 CK4J9W 44584852 IC50 = 2.6 nM T13453 C0GTZ7 44587983 Ki = 160 nM T13453 C20WUX 44587984 Ki = 51.5 nM T13453 CGU02F 54764328 IC50 = 380 nM T13453 CD87IE 54764411 IC50 = 330 nM T13453 CPZ93G 54764412 IC50 = 380 nM T13453 C1TO0M 57390716 IC50 = 770 nM T13453 CKE01G 57390718 IC50 = 24850 nM T13453 C32ETJ 57392517 IC50 = 1060 nM T13453 CR25FK 57392518 IC50 = 1930 nM T13453 C7P8NA 57394235 IC50 = 3380 nM T13453 C7AT3L 57394236 IC50 = 930 nM T13453 CY5D0W 57394237 IC50 = 1750 nM T13453 CJ39YQ 57394238 IC50 = 560 nM T13453 C0WBK1 57394239 IC50 = 540 nM T13453 C16SNJ 57394240 IC50 = 430 nM T13453 C8G4OA 57394241 IC50 = 4180 nM T13453 CR7Z6D 57394303 IC50 = 4570 nM T13453 CN0MS2 57394304 IC50 = 6620 nM T13453 COJ7T1 57395992 IC50 = 8650 nM T13453 CU6K8A 57395993 IC50 = 12500 nM T13453 CU93SZ 57395994 IC50 = 2080 nM T13453 CCEG86 57395995 IC50 = 980 nM T13453 CB70EI 57396058 IC50 = 1090 nM T13453 CD3FK9 57397796 IC50 = 3690 nM T13453 CI2RP0 57397797 IC50 = 8040 nM T13453 C7GK1B 57397798 IC50 = 1920 nM T13453 CD35FB 57397799 IC50 = 440 nM T13453 C2W0JH 57399456 IC50 = 3400 nM T13453 C2H3XW 57399457 IC50 = 550 nM T13453 CZ9RD1 57399458 IC50 = 2030 nM T13453 CR9WH3 57399459 IC50 = 780 nM T13453 CS27BV 57401220 IC50 = 4150 nM T13453 C8DS7R 57401221 IC50 = 770 nM T13453 CO40GM 57401222 IC50 = 1180 nM T13453 CIO4Q9 57401223 IC50 = 2850 nM T13453 CT7PZ3 57401225 IC50 = 1340 nM T13453 CG1J8I 57401228 IC50 = 9070 nM T13453 CYR89Z 71508528 Ki = 15.6 nM T13453 C0O3CM 71720536 Ki = 119 nM T13453 CWH6T3 72548703 IC50 = 0.19 nM T13453 D01LMH 25180489 Ki = 17.5 nM T13453 D02GOE 44563954 Ki = 16.1 nM T13453 D02JQP 24760995 Ki = 51.5 nM T13453 D03ECE 44563952 Ki = 14.9 nM T13453 D05GFD 44563953 Ki = 14.4 nM T13453 D06DWA 44563958 Ki = 20.5 nM T13453 D07NOJ 45104655 Ki = 35 nM T13453 D09SDZ 44587982 Ki = 13 nM T13453 D0DD3F 44563955 Ki = 18.2 nM T13453 D0EO5F 44563956 Ki = 51.5 nM T13453 D0H4DF 16132126 Ki = 1.1 nM T13453 D0H9QA 25180495 Ki = 48 nM T13453 D0PY7O 6324638 Ki = 1.74 nM T13453 D0Q3CB 16133821 Ki = 1.5 nM T13453 D0S4VO 45104657 Ki = 20.2 nM T13453 D0TF7R 44563951 Ki = 24 nM T13453 D0V7UG 45104656 Ki = 15.9 nM T13453 D0Z3QG 44563957 Ki = 15 nM T89530 CW9G5L 150570 IC50 = 2170 nM T89530 C4QG8H 3508054 IC50 = 50 nM T89530 C0U6YX 3508059 IC50 = 1250 nM T89530 CMA40L 5092911 IC50 = 31700 nM T89530 CKP1Y4 90644339 IC50 > 100000 nM T89530 CYD71G 90644340 IC50 = 980 nM T89530 CMXY84 90644341 IC50 = 11800 nM T89530 CFVS82 90644342 IC50 = 15840 nM T89530 C2QDT0 90644343 IC50 = 13100 nM T89530 C8CXG2 90644344 IC50 = 5210 nM T89530 CHM46Z 90644345 IC50 = 660 nM T89530 CGM5N0 90644346 IC50 = 430 nM T89530 CM2J0G 90644347 IC50 = 2010 nM T89530 CL7CK6 90644348 IC50 = 33850 nM T89530 CS0AD6 90644349 IC50 = 210 nM T89530 C14GOM 90644350 IC50 = 180 nM T89530 C8GR5L 90644351 IC50 = 35400 nM T89530 C9OZ5L 90644352 IC50 > 100000 nM T89530 CLQ0C1 90644353 IC50 = 41990 nM T89530 CKL0B7 90644354 IC50 > 100000 nM T89530 CK31VW 90644355 IC50 = 31800 nM T89530 CET02U 90644356 IC50 = 180 nM T89530 C2I1VP 90644357 IC50 = 90 nM T89530 C8X9UO 90644358 IC50 = 140 nM T89530 CA7EU1 90644359 IC50 = 110 nM T89530 C7DPQ0 90644360 IC50 = 40 nM T89530 CZU1J4 90644361 IC50 = 3040 nM T89530 C4F6ZI 90644362 IC50 = 1090 nM T89530 CA21TC 90644363 IC50 = 730 nM T89530 CRL8E2 90644364 IC50 = 1350 nM T89530 C4E6WO 90644365 IC50 = 50900 nM T89530 CV76KR 90644366 IC50 = 22100 nM T03403 D03RTS 2662 IC50 = 89 nM T03403 D0GY5Z 2244 IC50 = 15000 nM T03403 D0R1RS 3715 IC50 = 10 nM T03403 D0U2FN 71321 IC50 = 6500000 nM T03403 D05WPQ 6438354 IC50 = 3200 nM T03403 D09QRO 55390 IC50 = 10000 nM T03403 D0DP8P 47795 IC50 = 5800 nM T03403 D0JY4Y 443292 IC50 > 100000 nM T03403 D0N1SU 133021 IC50 = 160 nM T03403 D0O8ZE 5059 IC50 = 5300 nM T03403 D0S8YL 3969 IC50 = 44000 nM T03403 CH0L7P 71697 IC50 = 950000 nM T03403 CI5D9O 92656 IC50 = 100 nM T03403 CV7L0G 112230 IC50 = 100000000 nM T03403 CT2XZ0 116545 IC50 = 7079457.84 nM T03403 CAT4E3 129615 IC50 = 3388441.56 nM T03403 CCJ76H 512829 IC50 = 9000 nM T03403 CE2BC3 512830 IC50 = 14000 nM T03403 C16VBD 512831 IC50 = 12000 nM T03403 CT7E6Y 573683 IC50 > 800000 nM T03403 CZ0AH3 638278 IC50 = 130000 nM T03403 C6EVL8 854057 IC50 = 3467368.5 nM T03403 CQM64G 3037018 IC50 = 800 nM T03403 COH1C4 3052566 IC50 = 446683.59 nM T03403 C82IPJ 3052567 IC50 = 912010.84 nM T03403 C4VBK3 3253091 IC50 = 50000 nM T03403 CU86JL 4618600 IC50 = 40000 nM T03403 C4M1JC 5709318 IC50 = 44000 nM T03403 COQ7T3 5973690 IC50 = 63000 nM T03403 C3G7DT 6365297 IC50 = 4200 nM T03403 C40FZG 6366698 IC50 = 1300 nM T03403 C02AQY 6366699 IC50 ~ 1000 nM T03403 CWK1F9 6438990 IC50 = 110 nM T03403 C62UOZ 6439221 IC50 = 780 nM T03403 CHQ4Z3 6439222 IC50 = 1300 nM T03403 COC86Q 6439421 IC50 = 390 nM T03403 CLJ91K 6439912 IC50 = 260 nM T03403 C82TEX 7515046 IC50 < 10000 nM T03403 CUS6L8 9822795 IC50 = 30 nM T03403 C5C9ET 10042219 IC50 > 100000 nM T03403 C9T7YV 10063338 IC50 > 100000 nM T03403 CBL7R3 10220019 IC50 = 400 nM T03403 C2WE0I 10246235 IC50 = 9600 nM T03403 C20BTQ 10313997 IC50 = 5500 nM T03403 C8EQI3 10334136 IC50 > 100000 nM T03403 CC1UF0 10335738 IC50 > 100000 nM T03403 C25MYB 10425738 IC50 > 100000 nM T03403 CPR7J0 10469807 IC50 = 12589254.12 nM T03403 C6JI5F 10492615 IC50 > 300000 nM T03403 C0NRO9 10513373 IC50 = 570000 nM T03403 CK0OL2 10704667 IC50 = 27000 nM T03403 CUOI16 10729548 IC50 = 26000 nM T03403 C8IBM2 10801359 IC50 = 250000 nM T03403 CC8S6O 10801786 IC50 = 37000 nM T03403 CDZ94R 10826230 IC50 = 29000 nM T03403 CGLQ72 11723348 IC50 > 100000 nM T03403 CH9VC8 13245625 IC50 > 10000 nM T03403 CRA87I 13556944 IC50 = 14125375.45 nM T03403 C0P5AK 13914227 IC50 > 100000 nM T03403 C49OGE 13914253 IC50 > 100000 nM T03403 C4U3RD 14006855 IC50 = 5000 nM T03403 C6EZ0K 14312565 IC50 > 10000 nM T03403 C2X8PQ 14416570 IC50 = 34 nM T03403 C5PT1G 14416572 IC50 670 nM T03403 C1SG0F 14416576 IC50 = 10000 nM T03403 CRYI80 14416580 IC50 = 610 nM T03403 C27NOS 14416585 IC50 < 10000 nM T03403 C6BP2F 14416587 IC50 < 1000 nM T03403 CER87K 14762923 IC50 = 13803842.65 nM T03403 CGYF09 14762938 IC50 = 501187233.6 nM T03403 CX9AH8 14762939 IC50 = 501187233.6 nM T03403 CU3OT4 14762940 IC50 = 165958690.7 nM T03403 CXT3B5 14762942 IC50 = 100000000 nM T03403 CNZ45J 14762943 IC50 = 91201083.94 nM T03403 CL2A1E 14762944 IC50 = 91201083.94 nM T03403 C78IHC 14762948 IC50 = 50118723.36 nM T03403 CBL2O8 14762951 IC50 = 14791083.88 nM T03403 C8NKZ7 14762954 IC50 = 7079457.84 nM T03403 C4PS0F 14771889 IC50 < 10000 nM T03403 CV41BE 14771890 IC50 = 3100 nM T03403 CCX7K5 14771891 IC50 = 1400 nM T03403 CG57JP 14771892 IC50 = 1300 nM T03403 C91VJM 14771893 IC50 = 230 nM T03403 C0EMA5 14771894 IC50 < 1000 nM T03403 CZ4WJ2 14771895 IC50 = 730 nM T03403 CV5YH8 14771896 IC50 < 10000 nM T03403 C3HNQ2 14771897 IC50 < 10000 nM T03403 CH0TC9 14771898 IC50 < 10000 nM T03403 CX3N7Z 14771899 IC50 = 11000 nM T03403 CX7VA0 14771900 IC50 < 10000 nM T03403 CZC2D4 14771901 IC50 < 10000 nM T03403 CTY60Q 14771902 IC50 < 10000 nM T03403 C0D5OC 14771903 IC50 = 1500 nM T03403 CS3V5C 14771904 IC50 < 10000 nM T03403 CNH5M1 14771905 IC50 = 3200 nM T03403 CXN94C 14771906 IC50 = 510 nM T03403 CY2HF8 14771907 IC50 = 1400 nM T03403 CP5M9A 14771908 IC50 = 190 nM T03403 CI3XK7 14771909 IC50 < 10000 nM T03403 C8NTK2 14771910 IC50 = 750 nM T03403 C8H6XA 14771911 IC50 = 2500 nM T03403 CK53TR 14771912 IC50 < 1000 nM T03403 C10DIY 14771913 IC50 < 1000 nM T03403 C2F9TX 14771915 IC50 = 1100 nM T03403 C83VPQ 14771916 IC50 = 710 nM T03403 CA0C7U 14771917 IC50 = 1000 nM T03403 CK0AR5 14771918 IC50 < 1000 nM T03403 C8SRH6 14771919 IC50 > 10000 nM T03403 CCS9Y4 14771920 IC50 > 10000 nM T03403 C47LJK 14771921 IC50 > 10000 nM T03403 C9OWP0 14771922 IC50 = 1300 nM T03403 C1Z6FX 14771923 IC50 = 780 nM T03403 CHI8M3 14771924 IC50 < 10000 nM T03403 C4JX5S 14771927 IC50 = 590 nM T03403 CRGJ45 14771928 IC50 < 10000 nM T03403 C7L2ZJ 14771929 IC50 = 400 nM T03403 CXAG49 14771930 IC50 < 1000 nM T03403 C54ITL 14771931 IC50 = 110 nM T03403 CC4LM1 14771932 IC50 < 10000 nM T03403 CU6TO3 14771933 IC50 < 10000 nM T03403 C08CRZ 14771934 IC50 = 630 nM T03403 CA3D5U 14771935 IC50 = 1000 nM T03403 CZU2H5 14771936 IC50 = 300 nM T03403 C3B0LX 14771937 IC50 < 10000 nM T03403 CRT9E4 14771938 IC50 > 10000 nM T03403 C18DXV 14977360 IC50 = 71000 nM T03403 CD8YK4 15256755 IC50 = 140000 nM T03403 C53TQI 19044744 IC50 > 100000 nM T03403 CGPW68 19044748 IC50 > 100000 nM T03403 CLN6S5 19044753 IC50 > 100000 nM T03403 CR1W2E 19934882 IC50 > 100000 nM T03403 CF30ID 23275601 IC50 = 66069344.8 nM T03403 CUC36F 23680215 IC50 = 9772372.21 nM T03403 CN6F4H 23680216 IC50 = 4365158.32 nM T03403 C2JUV4 23680221 IC50 = 17782794.1 nM T03403 CHY73S 23680224 IC50 = 524807460.3 nM T03403 C7HV8Y 23680227 IC50 = 70794578.44 nM T03403 CZV8U1 23680228 IC50 = 4677351.41 nM T03403 C54NWH 23680229 IC50 = 741310241.3 nM T03403 CNU43B 23680230 IC50 = 891250938.1 nM T03403 C8A9UV 23689693 IC50 = 562341325.2 nM T03403 CJ1Z9S 44315480 IC50 = 794328234.7 nM T03403 C7UG4F 44315519 IC50 = 15135612.48 nM T03403 C8FEV0 44319113 IC50 = 25000 nM T03403 C1ZH6U 90664380 IC50 > 100000 nM T03403 C5T4EQ 131801158 IC50 = 23 nM T03403 C6JF0E 135616214 IC50 = 2500 nM T03403 CH4YE6 135987613 IC50 > 10000 nM T03403 CFNO28 145950339 IC50 = 34 nM T03403 CG37FR 145950583 IC50 = 27 nM T03403 CCN16Y 145952805 IC50 = 44 nM T03403 C2FVO7 145953074 IC50 = 38 nM T03403 C19TPY 145958203 IC50 = 50 nM T03403 C1BLR8 145959460 IC50 = 33 nM T03403 CUXQ13 145971245 IC50 = 41 nM T03403 C8U9TX 145971276 IC50 = 28 nM T03403 D00GBX 71751 IC50 = 5.7 nM T03403 D01TOR 667555 IC50 = 50000 nM T03403 D05EMX 14076674 IC50 = 10000000 nM T03403 D06VWH 11758240 IC50 = 2 nM T03403 D08GOT 13752584 IC50 = 4897788.19 nM T03403 D09AUL 10266864 IC50 = 51000 nM T03403 D0EW3L 5281222 IC50 = 120000 nM T03403 D0M6UM 129265 IC50 = 22000 nM T03403 D0P1LP 7090 IC50 = 12000 nM T03403 D0U0YE 14762941 IC50 = 165958690.7 nM T03403 D0U2YL 131820 IC50 = 36000 nM T03403 D0U8YQ 921562 IC50 = 14000 nM T37417 D0E3TC 44259 IC50 = 1.47 nM T37417 CV63UL 67240318 IC50 > 10000 nM T37417 C2MD1Q 155513187 IC50 > 10000 nM T83193 D03LGG 1548942 EC50 = 28.2 nM T83193 D05JNI 8378 IC50 = 400 nM T83193 D07ILQ 4671 EC50 > 10000 nM T83193 D0BQ8Y 5971 EC50 = 160000 nM T83193 D0U5CE 1548943 EC50 = 2.512 nM T83193 D00CMV 11256560 IC50 = 0.7 nM T83193 D05XJW 5702546 EC50 = 0.019 nM T83193 D07AOL 16741 EC50 = 180000 nM T83193 D0CO6D 71144018 IC50 > 20000 nM T83193 D0EM4S 17751090 IC50 = 4.6 nM T83193 D0H7PW 638024 EC50 = 3162.28 nM T83193 D07LRT 8068410 IC50 = 2.1 nM T83193 D07EAV 66644203 Ki = 0.04 nM T83193 D09ZWU 66644325 Ki = 0.1 nM T83193 D0K3KE 24782891 IC50 = 25 nM T83193 D0NV2M 52949700 IC50 = 130 nM T83193 D0ZM8H 25265637 IC50 = 34 nM T83193 D0L5XI 16007367 IC50 = 0.6 nM T83193 D0VJ5N 9910486 IC50 = 100 nM T83193 D0Z0PB 11247522 IC50 = 1.1 nM T83193 CT3IS2 2346 EC50 = 223000 nM T83193 CNG85F 3473 EC50 = 3300 nM T83193 C1MO7R 8842 IC50 > 100000 nM T83193 CU94MR 9017 IC50 > 100000 nM T83193 C76SDU 75263 EC50 = 100000 nM T83193 C7UD3V 78151 EC50 = 100000 nM T83193 CTEY14 160611 EC50 = 170000 nM T83193 CF7G0R 160785 EC50 = 1.995 nM T83193 C0GD6Q 310417 IC50 = 3.5 nM T83193 C2QKN6 441539 EC50 = 26000 nM T83193 CE51PH 581676 EC50 = 6309.57 nM T83193 C8WO2M 609524 EC50 = 390 nM T83193 C37RCW 622545 EC50 = 6600 nM T83193 CI9TY8 641115 EC50 = 19952.62 nM T83193 CFMR42 641296 IC50 > 10000 nM T83193 CIX6Q2 643820 IC50 > 100000 nM T83193 C7JSO8 667594 IC50 = 270 nM T83193 CUN5Q0 671605 EC50 > 10000 nM T83193 CFZ3U9 677890 IC50 = 7100 nM T83193 C1YV5I 680436 IC50 = 140 nM T83193 CJ5HC3 692312 IC50 > 10000 nM T83193 CB6LT1 692324 IC50 > 10000 nM T83193 C0XD7N 692351 IC50 > 10000 nM T83193 CY0I3M 721917 IC50 = 147 nM T83193 CS61UR 723775 IC50 = 2500 nM T83193 C7INU2 727129 IC50 = 570 nM T83193 CV2R0I 732540 IC50 > 4000 nM T83193 C2RJ1B 749814 IC50 = 550 nM T83193 CYW3D8 766652 EC50 = 2700 nM T83193 CJD52G 790345 IC50 > 10000 nM T83193 C4M6AL 792621 IC50 = 10700 nM T83193 C5M0TR 871278 IC50 = 2100 nM T83193 CVL8W6 886896 IC50 = 1000 nM T83193 CPED72 887195 IC50 = 210 nM T83193 CVX97S 924972 IC50 > 10000 nM T83193 CY71JK 985818 IC50 > 10000 nM T83193 CR37XU 1245920 IC50 > 10000 nM T83193 CC5NZ4 1322679 IC50 = 320 nM T83193 CC0SH7 1549025 IC50 > 100000 nM T83193 CZ9UX2 1549026 IC50 > 100000 nM T83193 C6UK7A 2093845 IC50 = 210 nM T83193 COZ7X0 2163913 IC50 = 370 nM T83193 C3W6KF 2165451 IC50 > 10000 nM T83193 CD2U7F 2176913 IC50 = 190 nM T83193 CY2U4R 2272103 IC50 > 10000 nM T83193 CC1B7S 2671351 IC50 > 10000 nM T83193 C37EXF 2684177 IC50 > 10000 nM T83193 CG4N3Y 2773243 IC50 > 10000 nM T83193 C6TFN7 3024586 EC50 = 12.59 nM T83193 CN7L2E 3312764 EC50 = 700 nM T83193 CM62BA 3684843 IC50 = 3.9 nM T83193 CY2FP6 4169432 IC50 = 4230 nM T83193 C7WX8B 4391297 IC50 = 7350 nM T83193 CU6M8E 5280457 IC50 > 10000 nM T83193 CJ7NK6 5281719 IC50 = 15000 nM T83193 CZM7D8 5281794 EC50 = 320 nM T83193 CHL79T 5282363 IC50 > 10000 nM T83193 C1UI3F 5283663 IC50 = 1400 nM T83193 C2F8DE 5284650 IC50 > 10000 nM T83193 CA95OR 5311093 EC50 = 0.5012 nM T83193 CZ46HG 5315659 EC50 = 1300 nM T83193 CQM1P0 5316874 IC50 > 10000 nM T83193 C1RM8Q 5317148 IC50 = 5000 nM T83193 C14GJD 5320618 EC50 = 3981.07 nM T83193 CWAE41 5320621 EC50 = 6.31 nM T83193 CB1GY5 5330587 IC50 = 29 nM T83193 C5ZM8C 5330591 IC50 = 45 nM T83193 CETR65 5366045 EC50 = 4000 nM T83193 C3XA4D 5375465 IC50 > 10000 nM T83193 CU7MX6 5375953 IC50 > 10000 nM T83193 CLO2Q0 5375954 IC50 > 10000 nM T83193 CPX84Y 5394296 IC50 > 10000 nM T83193 C25YUO 5458190 EC50 = 20000 nM T83193 CVD3P2 5704872 IC50 > 10000 nM T83193 CX56UR 5704879 IC50 > 10000 nM T83193 C8JDF6 5775508 IC50 > 10000 nM T83193 CR9HU5 5795514 IC50 = 360 nM T83193 CQG8Z1 5930975 IC50 > 10000 nM T83193 CYU86S 5962587 IC50 > 10000 nM T83193 C6JTH9 6016362 IC50 > 10000 nM T83193 C61ZKG 6018729 IC50 > 4000 nM T83193 CIAL25 6029870 IC50 = 1800 nM T83193 CVC96K 6146604 IC50 = 21 nM T83193 CQ6W2K 6187443 IC50 = 82 nM T83193 C38SOC 6442187 IC50 > 10000 nM T83193 CH1ZX4 6445256 EC50 = 2511.89 nM T83193 CP6D9U 6450018 EC50 = 1.995 nM T83193 C3XYQ7 7354608 IC50 = 370 nM T83193 C1V8ZN 7825385 IC50 = 1200 nM T83193 C83PLM 7914251 IC50 = 120 nM T83193 CD9K5W 7926018 IC50 > 10000 nM T83193 C92YOX 8643775 IC50 = 3490 nM T83193 CVE26J 8668560 EC50 = 4620 nM T83193 CNWP54 8702029 IC50 = 46 nM T83193 C6QO1A 8763094 Ki = 400 nM T83193 C4BYR6 8802859 IC50 = 4100 nM T83193 CHD5I9 9191541 IC50 = 170 nM T83193 CIW52Q 9795270 EC50 = 1200 nM T83193 C8GA6Z 9800250 IC50 = 3.3 nM T83193 CW4Z5B 9802648 Ki = 1.2 nM T83193 CDSI92 9804872 Ki < 10 nM T83193 CY1IX4 9806014 EC50 = 1.34 nM T83193 CKDU64 9819027 Ki = 0.3 nM T83193 C9M0GR 9843337 EC50 = 21300 nM T83193 C7G4AN 9867739 Ki = 3 nM T83193 CS6FN7 9883254 IC50 > 30000 nM T83193 CZJV79 9885200 EC50 = 28100 nM T83193 C67XMD 9885883 EC50 = 22400 nM T83193 C91VSG 9892415 IC50 = 1627 nM T83193 CWXR69 9906556 IC50 = 28 nM T83193 C1QTI8 9950097 IC50 = 18 nM T83193 C79EXD 9950886 IC50 = 26.5 nM T83193 CC0NE7 9975006 IC50 = 24 nM T83193 C19YQR 9975762 IC50 = 10 nM T83193 CVA29T 9975827 Ki = 2.8 nM T83193 C7EK0F 9975828 Ki = 2 nM T83193 CELG21 9977590 IC50 = 3.8 nM T83193 CO7A0B 9983112 IC50 = 0.9 nM T83193 C5D3QA 9985117 IC50 = 0.5 nM T83193 CJ9VY2 9998549 IC50 = 19 nM T83193 C7RX8V 9998550 IC50 = 19 nM T83193 CC0KE3 10022547 IC50 = 15.5 nM T83193 CU02IO 10025997 EC50 = 3.981 nM T83193 C0GC4S 10027372 IC50 = 270 nM T83193 C2UHV7 10028367 Ki = 2 nM T83193 CF41ZU 10041746 IC50 = 680 nM T83193 C2K6IJ 10050089 IC50 = 4 nM T83193 CW29KD 10064626 Ki = 1110 nM T83193 CD84LG 10066181 IC50 = 4 nM T83193 CF4CJ3 10070949 IC50 = 200 nM T83193 CR93GP 10071063 Ki = 4 nM T83193 CB34HN 10084135 EC50 = 1100 nM T83193 CX1DC7 10089889 Ki = 1 nM T83193 C71NWR 10090630 EC50 = 0.5012 nM T83193 CHJB75 10090920 Ki = 1 nM T83193 CNU5H6 10097731 IC50 > 3000 nM T83193 C1RTO5 10125879 IC50 = 620 nM T83193 C8U6LR 10126213 IC50 = 210 nM T83193 C8FKH7 10127170 IC50 = 14 nM T83193 C0IRH4 10127277 IC50 = 7 nM T83193 C5GBZ9 10134409 IC50 = 2.2 nM T83193 CG7VD1 10137465 IC50 = 120 nM T83193 CPZ8N5 10149904 IC50 = 36 nM T83193 CF4Y2Q 10149955 IC50 = 170 nM T83193 C5UAW7 10151288 IC50 = 0.63 nM T83193 CA8J7D 10158754 IC50 = 3.4 nM T83193 CYL9Z3 10171348 IC50 > 10000 nM T83193 C4PA2N 10172003 EC50 = 440 nM T83193 CXT21K 10172112 IC50 = 110 nM T83193 CZRS09 10174189 IC50 = 25 nM T83193 CXRA70 10193842 IC50 = 58 nM T83193 C80JFQ 10194497 IC50 = 20 nM T83193 CHO90S 10194542 IC50 = 60 nM T83193 C30SET 10194869 IC50 = 15 nM T83193 CXOT69 10215278 IC50 = 960 nM T83193 C83KOY 10215307 IC50 = 57 nM T83193 CVR7Y5 10215323 IC50 = 100 nM T83193 C01ESY 10215461 IC50 = 6.5 nM T83193 CZV42N 10215462 IC50 = 270 nM T83193 CHL48Q 10216527 IC50 = 32 nM T83193 C84DFK 10237015 IC50 = 67 nM T83193 CR8W2O 10237016 IC50 = 33 nM T83193 CEB7X5 10238224 IC50 = 2.5 nM T83193 C46FGC 10238413 IC50 = 0.5 nM T83193 CI3CN0 10247042 IC50 = 5.3 nM T83193 CC5HS4 10248318 IC50 = 0.3 nM T83193 CX7UD3 10252323 EC50 = 3.162 nM T83193 CG42MQ 10254025 Ki = 20 nM T83193 CPY9C7 10255515 IC50 = 1015 nM T83193 C2O0AJ 10286990 IC50 = 360 nM T83193 CFL3R4 10288125 IC50 = 290 nM T83193 CCFL59 10291273 IC50 = 5.4 nM T83193 CU90PR 10296445 IC50 = 17 nM T83193 CUW8F6 10308903 IC50 = 2.5 nM T83193 CHXI91 10308951 IC50 = 100 nM T83193 CIGM15 10309581 IC50 = 16 nM T83193 CZ6AM2 10312273 IC50 = 8 nM T83193 CRJ50W 10317518 IC50 = 23.8 nM T83193 CP61TH 10320921 IC50 > 1000 nM T83193 C3HS0L 10322861 IC50 = 25 nM T83193 CJ30SL 10323420 IC50 = 380 nM T83193 CQG58D 10340730 IC50 = 156 nM T83193 C2PI9Q 10341359 Ki = 4 nM T83193 CJ3UF9 10344203 EC50 = 2.512 nM T83193 C0S8FJ 10344437 IC50 = 162 nM T83193 CZKJ20 10344725 Ki = 2 nM T83193 C3NQS1 10357804 Ki = 53 nM T83193 CSW7F0 10367774 IC50 = 1.5 nM T83193 C8DIR2 10382943 IC50 = 123 nM T83193 CC0WP2 10384501 IC50 = 26 nM T83193 C2JI8H 10385075 Ki = 0.8 nM T83193 CGP7U6 10385728 IC50 = 258 nM T83193 C9LFI6 10385845 IC50 = 2.8 nM T83193 CA1IV9 10386145 IC50 = 9.3 nM T83193 CYZG38 10387678 IC50 = 259 nM T83193 C3L9UM 10404960 IC50 = 143 nM T83193 CD2YP6 10406258 IC50 = 189 nM T83193 C29VNT 10406294 IC50 = 51 nM T83193 C6HQY1 10411678 IC50 = 392 nM T83193 CI9P1W 10425263 Ki > 10000 nM T83193 C13MQT 10425327 IC50 = 45 nM T83193 CEH01T 10426159 IC50 = 157 nM T83193 CI0JE6 10428579 Ki = 2.1 nM T83193 C57ZQU 10429018 IC50 = 3.7 nM T83193 CMG9A6 10429408 IC50 = 120 nM T83193 CWO2L8 10429507 IC50 = 3.3 nM T83193 C3LQN4 10447001 IC50 = 1000 nM T83193 CL8IZ5 10448190 IC50 = 6 nM T83193 CEQ06G 10450954 IC50 = 318 nM T83193 CBFE05 10451213 Ki = 1.3 nM T83193 C0U8LP 10452082 Ki = 6 nM T83193 CCAD19 10452485 Ki = 3280 nM T83193 CMPQ64 10452949 IC50 = 9.8 nM T83193 C4N1DL 10453522 IC50 = 0.4 nM T83193 CVFR67 10454306 Ki = 6 nM T83193 CYP0X1 10455072 IC50 = 93 nM T83193 C8AT1X 10455135 IC50 = 43 nM T83193 CV4J7H 10456001 Ki = 5 nM T83193 CAQF96 10472785 IC50 = 37 nM T83193 C25ZDB 10473617 IC50 = 22 nM T83193 CMK18G 10473758 EC50 > 4000 nM T83193 C6LOK4 10474580 Ki = 1 nM T83193 CBXL67 10478501 Ki = 2 nM T83193 C5P1KO 10873969 EC50 = 1.995 nM T83193 CI61XB 10914412 IC50 = 631 nM T83193 C2AHD6 10915682 IC50 = 251.6 nM T83193 C2J6TG 10919020 EC50 = 125.89 nM T83193 CA3B2H 10935516 EC50 = 794.33 nM T83193 CMQP95 10967355 EC50 > 100000 nM T83193 C2LN1R 10972111 EC50 = 6.31 nM T83193 C2VGU8 10974108 EC50 = 1.585 nM T83193 CJN8F0 11050348 EC50 = 501.19 nM T83193 CWE1X8 11081004 EC50 = 794.33 nM T83193 CFP20M 11081027 EC50 = 3.162 nM T83193 CS5FM3 11088005 EC50 = 39.81 nM T83193 C0JHT3 11111493 IC50 = 16.1 nM T83193 CVR3M4 11122626 IC50 = 126.2 nM T83193 CHU16K 11144513 EC50 = 1.259 nM T83193 CJ2FD9 11145177 EC50 = 79.43 nM T83193 C95ODG 11151251 EC50 = 7240 nM T83193 CFV06N 11152242 IC50 = 3 nM T83193 CDG10K 11154380 IC50 = 103 nM T83193 CPS86I 11154448 IC50 = 370 nM T83193 CLD61F 11154884 IC50 = 15 nM T83193 CI02FG 11162142 IC50 = 313 nM T83193 CP54RZ 11163439 IC50 = 3402 nM T83193 C6YWC5 11163678 IC50 = 489.5 nM T83193 CAE8L3 11164115 IC50 = 30 nM T83193 C1A4BU 11164323 IC50 = 21 nM T83193 CWM5V7 11169233 IC50 > 20000 nM T83193 CHY6X9 11174909 IC50 = 1.1 nM T83193 CAF06O 11176490 IC50 = 19 nM T83193 CXG1K0 11176566 IC50 = 104 nM T83193 C1J3LQ 11177997 IC50 = 27 nM T83193 C2SX3V 11185579 IC50 > 4000 nM T83193 CZL23J 11187009 IC50 = 11 nM T83193 C7RB6N 11187610 IC50 = 1500 nM T83193 CR4F1A 11201020 IC50 = 3900 nM T83193 C7M4GR 11202946 IC50 = 123 nM T83193 CM6I4W 11209975 IC50 = 987 nM T83193 CA7FV3 11210430 IC50 = 223 nM T83193 CW49IC 11210873 IC50 = 180 nM T83193 CHF3V9 11220874 IC50 = 68.2 nM T83193 C34WOG 11221698 IC50 = 42 nM T83193 C23SYW 11222319 IC50 = 618 nM T83193 C3XYU2 11233046 IC50 = 500 nM T83193 CU1FD5 11233174 IC50 = 33.4 nM T83193 C9VR3I 11234067 IC50 = 52.2 nM T83193 C6ZUV1 11234223 IC50 = 10 nM T83193 CF2AH5 11234438 IC50 = 124 nM T83193 CX8YP0 11234482 IC50 = 216 nM T83193 CJK04D 11234633 IC50 = 4.7 nM T83193 CGA41K 11235292 IC50 = 44 nM T83193 CZI71C 11235331 IC50 > 4000 nM T83193 CYW2F0 11235811 IC50 = 5030 nM T83193 CZ6MK4 11244984 IC50 = 6 nM T83193 CLOA71 11245391 EC50 = 1930 nM T83193 CR0K5D 11246068 IC50 > 10000 nM T83193 C97YAJ 11246431 IC50 = 3 nM T83193 C2NHQ7 11247081 IC50 = 708 nM T83193 CNW9A3 11247815 IC50 = 41 nM T83193 CKY53N 11255817 IC50 = 30 nM T83193 CKQ1P7 11256604 IC50 = 1220 nM T83193 CT2YA8 11257635 IC50 = 149 nM T83193 C9OWF3 11258604 EC50 > 10000 nM T83193 C6TY2P 11259004 IC50 > 538 nM T83193 CVC36Y 11266760 IC50 = 11 nM T83193 C8YO3L 11266761 IC50 = 46 nM T83193 C5WV4D 11267528 IC50 = 113 nM T83193 C0MJ8A 11268050 IC50 = 33 nM T83193 C56VSC 11268075 IC50 = 10 nM T83193 CR67LW 11278186 IC50 = 595 nM T83193 C9PM7U 11278403 IC50 = 110 nM T83193 C5OPQ9 11279403 IC50 = 87 nM T83193 CM08NB 11280561 IC50 = 170 nM T83193 CX5KL6 11281475 IC50 = 2746 nM T83193 CP5C7W 11281498 IC50 = 965 nM T83193 CH09YB 11290223 IC50 = 40 nM T83193 C5YH7T 11302584 IC50 > 4000 nM T83193 C8W2XI 11313411 IC50 = 10 nM T83193 CNP4Y7 11314287 IC50 = 9.8 nM T83193 CRK15B 11314719 IC50 = 223 nM T83193 CCR10K 11314913 IC50 = 3932 nM T83193 CMV01G 11317360 IC50 = 2700 nM T83193 C50RTJ 11325962 IC50 = 420 nM T83193 C6C5LA 11327231 Ki = 5.1 nM T83193 CU4QC7 11336651 IC50 = 2700 nM T83193 CN75HL 11337328 Ki = 8 nM T83193 CGR09J 11338019 IC50 = 14.2 nM T83193 CMV8T4 11338988 IC50 = 8 nM T83193 C02ELK 11348681 IC50 = 9544 nM T83193 CKD69Y 11360480 IC50 = 44 nM T83193 CD75ZO 11361213 IC50 = 1106 nM T83193 C1N5ED 11371933 IC50 = 2170 nM T83193 CU42XZ 11382833 IC50 = 10 nM T83193 CXO96B 11385287 IC50 = 2290 nM T83193 C8GJB1 11394405 IC50 = 1700 nM T83193 CID3X4 11394918 IC50 = 2415 nM T83193 CTK70N 11395736 IC50 = 15 nM T83193 C74LAW 11407011 IC50 = 6 nM T83193 C1C3TU 11407205 IC50 > 4000 nM T83193 CPU95G 11417553 IC50 = 52.3 nM T83193 CU7K1P 11420211 IC50 = 24 nM T83193 CDCB15 11426745 IC50 = 7200 nM T83193 CM15FO 11427765 IC50 = 150 nM T83193 CQTU13 11428484 IC50 = 290 nM T83193 CVL36R 11428656 IC50 = 270 nM T83193 CHZ75W 11428814 IC50 = 14 nM T83193 CQ13YN 11428847 IC50 = 58 nM T83193 CS2T0N 11430023 IC50 = 3 nM T83193 CE1IT2 11430396 IC50 = 64 nM T83193 CF9L0T 11439510 IC50 = 870 nM T83193 C4VDM3 11440418 IC50 > 4000 nM T83193 CEA7J0 11450944 IC50 = 5030 nM T83193 CD2Z3V 11451387 IC50 = 8 nM T83193 CB6O9N 11452823 IC50 = 3 nM T83193 C52AIL 11461948 IC50 = 3.7 nM T83193 CXC70P 11462535 IC50 = 3 nM T83193 CAW37B 11472797 IC50 = 27 nM T83193 C4J2HQ 11474026 IC50 = 78 nM T83193 CYUZ38 11474160 IC50 = 10 nM T83193 CP1KU4 11475509 IC50 = 44 nM T83193 C9M3QB 11476347 IC50 = 2450 nM T83193 C8XPK4 11484937 IC50 = 39 nM T83193 CRZ3D9 11485402 IC50 = 35 nM T83193 CN83SF 11486920 IC50 = 3383 nM T83193 CFU6A1 11487127 IC50 = 0.42 nM T83193 C07VMY 11494816 IC50 = 7 nM T83193 CM57GQ 11501549 IC50 = 670 nM T83193 C4YA8N 11501768 Ki = 125 nM T83193 CS3Z5T 11502982 IC50 = 29 nM T83193 CI9GW3 11510499 IC50 = 12 nM T83193 CQEK72 11515763 IC50 > 10000 nM T83193 C79ENI 11516347 IC50 = 43 nM T83193 CAVJ68 11516428 Ki = 314 nM T83193 CT30ZK 11516588 IC50 = 1070 nM T83193 CRL9B2 11516653 IC50 = 15 nM T83193 CY8JX7 11523773 IC50 = 1420 nM T83193 CKTQ89 11531155 IC50 = 230 nM T83193 CN6MQ9 11539037 IC50 = 1960 nM T83193 CWQ98U 11539631 Ki = 81 nM T83193 C08RMS 11545784 IC50 = 100 nM T83193 CJ0Y6C 11545915 Ki = 49 nM T83193 CL1DZ9 11545976 IC50 = 90 nM T83193 CDN4L6 11553027 IC50 = 70 nM T83193 CL6FO4 11554008 IC50 = 80 nM T83193 CVWG03 11560077 Ki = 93 nM T83193 C5CJ9Z 11566168 IC50 = 85.9 nM T83193 CB52VF 11566529 IC50 = 417.2 nM T83193 CXZG40 11568188 IC50 = 5610 nM T83193 CGZ52T 11568686 IC50 = 121 nM T83193 CDO0W8 11576806 IC50 = 870 nM T83193 C5ZA9N 11581212 IC50 = 46.7 nM T83193 CG2U8H 11581455 IC50 = 85.6 nM T83193 CV7KX2 11581829 Ki = 56 nM T83193 CMR49W 11582496 Ki = 65 nM T83193 C0BDS3 11588638 IC50 = 3 nM T83193 CS6G2H 11588890 IC50 = 4 nM T83193 CS5F7M 11594915 IC50 = 215 nM T83193 CG0L6V 11595037 IC50 = 1605 nM T83193 C4Z5JK 11595264 IC50 = 34 nM T83193 CDFN62 11595736 Ki = 225 nM T83193 CZ98PT 11601992 IC50 = 175.4 nM T83193 CYI2Z6 11603236 IC50 = 5 nM T83193 CZH2Y9 11610007 IC50 = 11.9 nM T83193 CI3RN0 11610880 Ki = 78 nM T83193 CSW1P8 11611379 IC50 = 66 nM T83193 C74UBE 11618868 IC50 = 800 nM T83193 C21AFU 11624859 Ki = 84 nM T83193 CZ60XH 11633359 Ki = 71 nM T83193 C6ET3R 11638123 IC50 = 234 nM T83193 C91TKC 11639553 IC50 = 41 nM T83193 C19YGI 11639605 Ki = 97 nM T83193 C0ZA2O 11646277 IC50 = 43 nM T83193 CHG1B2 11653471 IC50 = 5 nM T83193 CUDY54 11653760 Ki = 28 nM T83193 CJ15HT 11654024 IC50 = 8 nM T83193 CTD74A 11654160 IC50 = 6 nM T83193 CDZX61 11658617 EC50 = 115000 nM T83193 CB91CF 11661499 IC50 = 13 nM T83193 CD8EV7 11666821 EC50 = 600 nM T83193 CEC8W5 11668297 IC50 = 5 nM T83193 CJD1Q7 11668509 IC50 = 2871 nM T83193 CB0EI8 11669102 IC50 = 160 nM T83193 CIJD47 11674719 IC50 = 1810 nM T83193 CI9AN4 11675434 IC50 > 9000 nM T83193 CH04KW 11682087 IC50 = 19 nM T83193 CC2XH5 11682182 IC50 = 1688 nM T83193 C1QK7U 11688977 IC50 = 157 nM T83193 CHX6L1 11690649 IC50 = 8.4 nM T83193 C4AV3B 11696122 IC50 = 1072 nM T83193 CX6GH9 11696727 Ki = 137 nM T83193 C9QY1C 11696849 IC50 = 110 nM T83193 CFD2G5 11696967 IC50 = 600 nM T83193 CA83LO 11697246 IC50 = 11 nM T83193 CR49WU 11697696 IC50 > 9000 nM T83193 CQSV96 11704438 Ki = 68 nM T83193 CFPJ48 11704662 IC50 = 330 nM T83193 CPW83D 11709865 IC50 > 10000 nM T83193 C0YRW3 11711740 IC50 = 196 nM T83193 CB98GN 11717565 Ki = 61 nM T83193 C0UD1M 11718030 IC50 = 5575 nM T83193 CWV86L 11718098 IC50 = 16 nM T83193 C07CUH 11719337 IC50 = 5 nM T83193 CQ5K8J 11724001 Ki = 7 nM T83193 CHEX57 11725098 IC50 = 11 nM T83193 C8GL3E 11727340 EC50 = 3.162 nM T83193 CB2Q0P 11732417 EC50 = 1.259 nM T83193 CZN6Q7 11738421 IC50 = 52 nM T83193 CMBH71 11739242 IC50 = 670 nM T83193 C0NKI6 11739244 IC50 = 10970 nM T83193 C6VAE8 11739513 Ki = 1.3 nM T83193 CV5TK7 11740163 Ki = 581 nM T83193 CSB74R 11740932 Ki = 85 nM T83193 CBYF51 11749185 IC50 = 5 nM T83193 CT8JR0 11749393 IC50 = 175 nM T83193 C3KOH6 11750331 IC50 = 78 nM T83193 CNI40X 11750583 IC50 = 4 nM T83193 CNK13I 11750695 IC50 = 9 nM T83193 CN3XY8 11755886 IC50 = 2 nM T83193 C9NIB4 11759242 IC50 = 50.3 nM T83193 C5W8VO 11771660 IC50 > 4000 nM T83193 CMU4J6 11772590 IC50 = 280 nM T83193 C4HG5M 11772885 IC50 = 1100 nM T83193 CFB1Z4 11833616 EC50 = 199.53 nM T83193 C1DA0K 11951378 IC50 = 1.4 nM T83193 CCS69F 11951545 IC50 = 1.1 nM T83193 CTY37U 11951546 IC50 = 1.1 nM T83193 C2J7CO 11951910 IC50 = 0.62 nM T83193 CA3BL2 11951911 IC50 = 0.65 nM T83193 C8FJ0P 11955840 IC50 = 374 nM T83193 CV4OB6 11964241 IC50 = 327 nM T83193 CG1D8J 11964255 IC50 = 8.3 nM T83193 CIB79J 11964256 IC50 = 26 nM T83193 CJ3K6G 11964259 IC50 = 15 nM T83193 C2AP5B 11964260 IC50 = 101 nM T83193 C0ZFA2 11964262 IC50 = 62 nM T83193 C6S3AR 11964282 IC50 = 81 nM T83193 C3G2IB 11964283 IC50 = 187 nM T83193 CPM18J 11964284 IC50 = 416 nM T83193 CD6Z2K 11964285 IC50 = 157 nM T83193 C5BG8I 11964318 IC50 = 1820 nM T83193 C3ZXI9 11964319 IC50 = 277 nM T83193 CV3RW9 12110672 EC50 = 30000 nM T83193 CE38OM 12444907 IC50 = 200000 nM T83193 C6VR2A 13309825 EC50 = 60 nM T83193 C7ENX9 13559595 EC50 = 2.512 nM T83193 CBD2C4 13989871 IC50 = 17490 nM T83193 CD6N1T 14954814 IC50 > 10000 nM T83193 C08CSK 16007091 IC50 = 7.943 nM T83193 C2UML7 16035164 IC50 = 42 nM T83193 CPCZ62 16040329 IC50 > 10000 nM T83193 C5CJ0D 16045350 IC50 = 9120 nM T83193 C8Q6HW 16117762 IC50 > 10000 nM T83193 CP86RN 16117763 IC50 > 10000 nM T83193 CGDN09 16223445 Ki = 8.8 nM T83193 CKL25Q 16223447 Ki = 0.9 nM T83193 CZ2Q1X 16223604 Ki = 0.43 nM T83193 CFPN71 16223606 Ki = 1.3 nM T83193 C9I5RW 16223607 Ki = 19.1 nM T83193 C74WGS 16223608 Ki = 0.2 nM T83193 CB76QU 16223640 Ki = 0.3 nM T83193 CBC1R8 16223641 Ki = 0.5 nM T83193 CQ8MY6 16223642 Ki = 0.29 nM T83193 COS90Q 16223643 Ki = 1.1 nM T83193 C56AXM 16223644 Ki = 0.2 nM T83193 CVF6K8 16223645 Ki = 1.4 nM T83193 CH2ZC4 16223802 Ki = 2.1 nM T83193 CX8BV1 16223803 Ki = 0.4 nM T83193 C1RSQ8 16223806 Ki = 7.2 nM T83193 C1TOC0 16223839 Ki = 39.2 nM T83193 CAH18B 16223840 Ki = 9.1 nM T83193 CW7HQ6 16223841 Ki = 0.2 nM T83193 C7KM4H 16223842 Ki = 0.7 nM T83193 CE37HV 16223843 Ki = 0.9 nM T83193 COF9C5 16223844 Ki = 14 nM T83193 C3XHC6 16223998 Ki = 1 nM T83193 CQOF10 16224035 Ki = 0.02 nM T83193 CPL04S 16224036 Ki = 1 nM T83193 C3D1WU 16224037 Ki = 1.3 nM T83193 C6DNC7 16224038 Ki = 3.8 nM T83193 CRO21Z 16224039 Ki = 1.4 nM T83193 CU17TP 16224040 Ki = 3.5 nM T83193 CG3JR8 16224242 Ki = 0.9 nM T83193 C6ZGN2 16224243 Ki = 1.5 nM T83193 CT2E5Q 16224245 Ki = 0.8 nM T83193 C6QD9N 16224246 Ki = 59 nM T83193 CXC0I5 16224444 Ki = 5 nM T83193 CY54BU 16224445 Ki = 1.4 nM T83193 C76PDI 16224446 Ki = 0.6 nM T83193 CM6GV1 16224447 Ki = 4.2 nM T83193 C83EKL 16224449 Ki = 0.6 nM T83193 CQ24AK 16224638 Ki = 2.8 nM T83193 CX0G5W 16224639 Ki = 2 nM T83193 C07ASX 16224640 Ki = 3.4 nM T83193 C7YN2J 16224642 Ki = 1.3 nM T83193 CPS78U 16224643 Ki = 1.4 nM T83193 CHB3W0 16224833 Ki = 2.7 nM T83193 CHK78N 16224834 Ki = 1.2 nM T83193 CSA4V5 16224837 Ki = 6.1 nM T83193 C36QHN 16225030 Ki = 21.6 nM T83193 C7VM5G 16225031 Ki = 0.6 nM T83193 CL4UA3 16225032 Ki = 0.9 nM T83193 CG30SO 16225239 Ki = 1.1 nM T83193 C85JKQ 16225240 Ki = 54 nM T83193 C3S0GA 16225241 Ki = 42 nM T83193 C2T6CF 16225242 Ki = 32.7 nM T83193 CPVX56 16225243 Ki = 0.9 nM T83193 C81WVR 16225448 Ki = 0.9 nM T83193 C31LGV 16225451 Ki = 0.02 nM T83193 CNU8G3 16225452 Ki = 72.1 nM T83193 CZ12PD 16225453 Ki = 1.1 nM T83193 C4ZBD7 16225649 Ki = 0.6 nM T83193 CSR0J5 16225650 Ki = 0.8 nM T83193 CV1MH0 16225651 Ki = 2.4 nM T83193 CM5PT1 16225652 Ki = 0.7 nM T83193 CB0VG2 16225653 Ki = 0.3 nM T83193 CM4VX3 16225654 Ki < 1000 nM T83193 CF5AP8 16225855 Ki = 58 nM T83193 CJ5V2W 16225857 Ki = 9.2 nM T83193 CZ49PD 16389464 EC50 = 5888.44 nM T83193 CVD1R5 16655083 EC50 = 1.5 nM T83193 CQ3R0B 16747867 IC50 = 35.3 nM T83193 CHRA32 16747868 IC50 = 10.3 nM T83193 C6HF8Y 16748125 IC50 = 5.2 nM T83193 CJ7CV2 16748127 IC50 = 4.6 nM T83193 CR20DT 16748248 IC50 = 7360 nM T83193 CA5T8K 16748249 IC50 = 133 nM T83193 C94SBD 16748250 IC50 = 18 nM T83193 C2Q7FT 16748251 IC50 = 54.5 nM T83193 CA9GR3 16748252 IC50 = 43.2 nM T83193 CL2RP7 16748373 IC50 = 12.6 nM T83193 CPEG41 16748374 IC50 = 21.3 nM T83193 CAXZ17 16749111 EC50 > 4000 nM T83193 CVIT85 16749133 IC50 = 7.3 nM T83193 CST26C 16749136 IC50 = 9.3 nM T83193 C6TBH1 16749139 IC50 = 3.3 nM T83193 C1RJ3C 16749216 EC50 > 4000 nM T83193 CMF78C 16749217 EC50 > 4000 nM T83193 C3CY2E 16749218 EC50 > 4000 nM T83193 CJM80O 16749240 IC50 = 5.7 nM T83193 C2K7RW 16749243 IC50 = 14 nM T83193 CB13OV 16749244 IC50 = 190 nM T83193 C96BJP 16749324 EC50 > 4000 nM T83193 CMSA17 16749325 EC50 > 4000 nM T83193 C7U1NO 16749326 EC50 > 4000 nM T83193 C5YG7M 16749350 IC50 = 29.5 nM T83193 CLS61T 16749351 IC50 = 39.3 nM T83193 CMZ32J 16749352 IC50 = 58.8 nM T83193 C3W8DT 16749353 IC50 = 26.9 nM T83193 C0YS5E 16749354 IC50 = 20.4 nM T83193 CHA4N8 16749355 IC50 = 14.8 nM T83193 CWUP76 16749434 EC50 > 4000 nM T83193 CYHC97 16749435 EC50 > 4000 nM T83193 CP3AM6 16749438 IC50 = 1.9 nM T83193 CRQ73A 16749440 EC50 > 4000 nM T83193 CEJ56F 16749462 IC50 = 25.5 nM T83193 CG65CN 16749463 IC50 = 82 nM T83193 C9E4TJ 16749464 IC50 = 157 nM T83193 CI90SF 16749465 IC50 = 1850 nM T83193 CE8I4J 16749466 IC50 = 285 nM T83193 C2G7YQ 16749467 IC50 = 305 nM T83193 CZSC57 16749540 EC50 > 4000 nM T83193 C2EMH9 16749541 EC50 > 4000 nM T83193 CJ9D8L 16749542 EC50 > 4000 nM T83193 C2DK7L 16749543 EC50 > 4000 nM T83193 C4P5CU 16749544 EC50 > 4000 nM T83193 C8GVO1 16749545 EC50 > 4000 nM T83193 CR8EN6 16749565 IC50 = 902 nM T83193 C7AY3O 16749566 IC50 = 19.8 nM T83193 CBNQ43 16749567 IC50 = 29 nM T83193 CX05KR 16749568 IC50 = 22.4 nM T83193 C7EVJ4 16749569 IC50 = 19 nM T83193 CLN50R 17026579 IC50 = 2090 nM T83193 COL7M1 17421069 IC50 > 20000 nM T83193 CI73MC 17946552 IC50 > 10000 nM T83193 CSCY81 18229223 IC50 = 220 nM T83193 C0M4ZI 20090380 IC50 = 6300 nM T83193 CCR2N0 20807401 IC50 > 100000 nM T83193 C1G6OB 21404983 EC50 > 500000 nM T83193 CD6H7C 21598349 EC50 = 7000 nM T83193 CPJ06C 22030032 IC50 = 3 nM T83193 CS2H5P 22030052 IC50 = 0.3 nM T83193 CTI18S 22030066 IC50 = 0.4 nM T83193 CP40BJ 22030080 IC50 = 50 nM T83193 C5L7FA 22030144 IC50 = 24 nM T83193 C1UR9X 22030149 IC50 = 8 nM T83193 CC74QX 22030158 IC50 = 1.2 nM T83193 CZT0O2 22030173 IC50 = 12 nM T83193 CTU13R 22030183 IC50 = 6 nM T83193 C1HX4L 22030187 IC50 = 1 nM T83193 C7Y2SH 22030227 IC50 = 184 nM T83193 CRG70B 22030273 IC50 = 25 nM T83193 C6I7AP 22030278 IC50 = 35 nM T83193 C7O8AG 22030332 IC50 = 26 nM T83193 C8D4WK 22030340 IC50 = 2.1 nM T83193 C72FHC 22030363 IC50 = 2 nM T83193 C08ZUA 22030387 IC50 = 9 nM T83193 CMVA64 22030491 IC50 = 69 nM T83193 CDP5Y6 22030498 IC50 = 22 nM T83193 C0AS3O 22032592 IC50 = 19 nM T83193 CS9HJ7 22032616 IC50 = 94 nM T83193 CZRU05 22032622 Ki = 1.2 nM T83193 C17MCO 22032643 IC50 = 109 nM T83193 C6DGX1 22170442 IC50 = 0.8 nM T83193 C2W7TH 22258331 Ki = 0.8 nM T83193 CCG43N 22296670 IC50 = 141000 nM T83193 CR95GN 22337681 IC50 = 184 nM T83193 C3IEK4 23112208 IC50 = 350 nM T83193 CQ6XH2 23344732 IC50 = 320 nM T83193 C21YMA 23537063 IC50 = 62 nM T83193 C0B6WM 23537081 IC50 = 4.5 nM T83193 C9AI6U 23537111 IC50 = 25 nM T83193 CRF62A 23655242 IC50 = 41 nM T83193 CFK41Y 24106939 IC50 = 750 nM T83193 C2Z7MA 24749054 IC50 = 5250 nM T83193 CG0S9O 24749055 IC50 > 10000 nM T83193 CS3HD4 24749056 IC50 > 10000 nM T83193 C38RVI 24749057 IC50 > 10000 nM T83193 C3TRX4 24749058 IC50 > 10000 nM T83193 C5HCO9 24749162 IC50 = 470 nM T83193 C3L9PN 24749163 IC50 = 950 nM T83193 CJM71S 24749268 IC50 = 2570 nM T83193 CMNG82 24749269 IC50 > 10000 nM T83193 C7A1XM 24749272 IC50 = 2130 nM T83193 CM80VR 24749273 IC50 = 680 nM T83193 CU8EK4 24749373 IC50 = 240 nM T83193 C3FB1Y 24749374 IC50 = 430 nM T83193 CNVL17 24749375 IC50 = 3800 nM T83193 CI5P1B 24749376 IC50 = 2630 nM T83193 CWJ38Z 24749377 IC50 > 10000 nM T83193 CSD74Y 24749378 IC50 > 10000 nM T83193 C9F4CD 24749379 IC50 = 720 nM T83193 C5FJX1 24749485 IC50 > 10000 nM T83193 COY93F 24749486 IC50 > 10000 nM T83193 CAP1H6 24749487 IC50 = 2820 nM T83193 CC5Y4U 24749488 IC50 > 10000 nM T83193 CZ2H9N 24749489 IC50 > 10000 nM T83193 C6X1VD 24749490 IC50 > 10000 nM T83193 CI0L7N 24749586 IC50 = 2400 nM T83193 C6OXY3 24749587 IC50 > 10000 nM T83193 CHA2W7 24749588 IC50 > 10000 nM T83193 C4YU1Z 24749589 IC50 > 10000 nM T83193 CG32EF 24749590 IC50 > 10000 nM T83193 CG2E6O 24749591 IC50 > 10000 nM T83193 C2WF7Z 24749592 IC50 > 10000 nM T83193 CJ4E8Q 24749698 IC50 > 10000 nM T83193 CZ3TN1 24757992 IC50 = 300 nM T83193 CM8U7N 24758358 IC50 = 4.9 nM T83193 CIG1Z2 24758469 IC50 = 6 nM T83193 CAL0Z8 24758809 IC50 = 25 nM T83193 C8M2ZV 24758810 IC50 = 12 nM T83193 CHW1G2 24758811 IC50 = 140 nM T83193 CL1B4P 24758812 IC50 = 400 nM T83193 C9KHG4 24758813 IC50 = 40 nM T83193 CDQ6V0 24758928 IC50 = 2 nM T83193 CZ95VW 24758929 IC50 = 280 nM T83193 COS08A 24758930 IC50 = 210 nM T83193 CQLK06 24759035 IC50 = 10 nM T83193 CVI60T 24759038 IC50 = 120 nM T83193 C5ZB7W 24759039 IC50 = 45 nM T83193 C0D6BW 24759147 IC50 = 250 nM T83193 CSY3H1 24759484 IC50 = 76 nM T83193 C8QY4E 24759485 IC50 = 5.7 nM T83193 CWD7S2 24768191 Ki = 23 nM T83193 C7CNH2 24768197 IC50 = 147 nM T83193 CY02IF 24768198 IC50 = 125 nM T83193 CMC85W 24768199 IC50 = 171 nM T83193 CWY73R 24768200 IC50 = 46 nM T83193 CHL87D 24768201 IC50 = 20 nM T83193 CXO93T 24768202 IC50 = 17 nM T83193 CBMO21 24768204 IC50 = 31000 nM T83193 C9OL1G 24768205 IC50 = 15900 nM T83193 CUT5L4 24768206 IC50 = 476 nM T83193 CV31NY 24768207 IC50 = 287 nM T83193 C3NTZ4 24768208 IC50 = 47 nM T83193 CE27QX 24768209 IC50 = 248 nM T83193 CTQ1W2 24777535 IC50 = 19 nM T83193 C1NIH2 24777650 IC50 = 5 nM T83193 CF65KY 24777651 IC50 = 151 nM T83193 C03AVT 24777652 IC50 = 1350 nM T83193 C2Q4KN 24777657 IC50 = 127 nM T83193 C8IE1C 24777768 IC50 = 9 nM T83193 C63OSW 24777769 IC50 = 7 nM T83193 CTF76E 24777770 IC50 = 5 nM T83193 CYDV94 24777771 IC50 = 4 nM T83193 CV4E5Y 24777772 IC50 = 14 nM T83193 CBFM91 24777773 IC50 = 65 nM T83193 CVT9S0 24777889 IC50 = 5820 nM T83193 CE2I0G 24782892 IC50 = 188 nM T83193 CMN74Q 24782895 IC50 = 37 nM T83193 CUP61J 24783145 IC50 = 97 nM T83193 CT31VS 24783399 IC50 = 6160 nM T83193 C0NCS2 24783400 IC50 = 907 nM T83193 C7C9HL 24783403 IC50 = 6 nM T83193 C7D6JX 24783656 IC50 = 38 nM T83193 CL8T0V 24784683 IC50 = 361 nM T83193 C94OHQ 24784927 IC50 = 1450 nM T83193 CHYD03 24785963 IC50 = 2360 nM T83193 CB20PL 24795576 EC50 = 5000 nM T83193 CR40XN 24882612 IC50 = 23 nM T83193 C53HIK 24882754 IC50 = 2 nM T83193 CBW81E 24882793 IC50 = 5 nM T83193 CJN68G 24882876 IC50 = 13 nM T83193 CO7TH0 24882956 IC50 = 19 nM T83193 C75JOU 24882957 IC50 = 14 nM T83193 C1DQZ5 24882958 IC50 = 11 nM T83193 CFS9X6 24882959 IC50 = 21 nM T83193 CMV64G 24883004 IC50 = 23 nM T83193 CD6C5J 24883048 IC50 = 9 nM T83193 CRT08K 24883050 IC50 = 64 nM T83193 CI05FC 24883053 IC50 > 5000 nM T83193 CH0X7O 24883095 IC50 > 5000 nM T83193 C9K3MG 24883145 IC50 = 3 nM T83193 C0PUW7 24883305 IC50 = 63 nM T83193 C94XJC 24883307 IC50 = 12 nM T83193 CQKS73 24883308 IC50 = 59 nM T83193 C74BIP 24883353 IC50 = 3 nM T83193 CZRP90 24883354 IC50 = 41 nM T83193 CCN98Y 24883355 IC50 = 30 nM T83193 C7ODK0 24952932 IC50 = 101 nM T83193 C9YNW1 24952933 IC50 = 85 nM T83193 CRXY84 24970014 Ki = 3.79 nM T83193 CL0Q2W 25063516 Ki = 387 nM T83193 CJV2N6 25063517 Ki = 1.7 nM T83193 CGB14D 25063519 Ki = 0.2 nM T83193 C63HTY 25063555 Ki = 169 nM T83193 C2CLW4 25063559 Ki = 0.3 nM T83193 CUE06S 25063560 Ki = 0.6 nM T83193 CDIT59 25063596 Ki = 3.5 nM T83193 COCD41 25063598 Ki = 68.8 nM T83193 C6TSU3 25063599 Ki = 0.3 nM T83193 CZ6XV1 25063600 Ki = 0.9 nM T83193 CAZ23X 25063601 Ki = 6.4 nM T83193 C8CG5I 25063673 Ki = 2.3 nM T83193 CYIO54 25063675 Ki = 0.3 nM T83193 CF6O7A 25063709 Ki = 0.6 nM T83193 C16RAM 25063712 Ki = 59.4 nM T83193 CKQT89 25063747 Ki = 1.1 nM T83193 C0OTC3 25063748 Ki = 28.6 nM T83193 C0NUI7 25063787 Ki = 1.9 nM T83193 CV5JH8 25098503 Ki = 11.9 nM T83193 CSL79N 25098504 Ki = 55.5 nM T83193 CAW8P2 25102898 Ki = 0.1 nM T83193 CSG03M 25102901 Ki = 56.4 nM T83193 CCT35Q 25103505 Ki = 49.3 nM T83193 CN8X5E 25103635 Ki = 65.9 nM T83193 CV17BS 25103751 Ki = 49 nM T83193 C3JDL5 25103752 Ki = 62.5 nM T83193 C2C8ML 25103753 Ki = 65.7 nM T83193 C2X5RB 25103754 Ki = 1.3 nM T83193 CX2DO1 25103755 Ki = 124 nM T83193 C3G0BK 25104002 Ki = 7.5 nM T83193 CQ2BL0 25104247 Ki = 103 nM T83193 CT1MR7 25104361 Ki = 88.7 nM T83193 C90GAW 25104362 Ki = 42.9 nM T83193 C5XM0A 25104364 Ki = 3.4 nM T83193 C3PQ4U 25104478 Ki = 2.4 nM T83193 CM63CF 25104699 Ki = 1.1 nM T83193 CYA91N 25123379 Ki = 4.4 nM T83193 CB5LO8 25124040 Ki = 25 nM T83193 CXS51N 25124352 Ki = 0.9 nM T83193 CVM5H0 25124353 Ki = 0.7 nM T83193 CX6GR1 25124356 Ki = 9.6 nM T83193 C6K7FP 25141397 IC50 = 3000 nM T83193 CXT31S 25147549 IC50 = 15 nM T83193 CG5SI9 25181624 IC50 = 118 nM T83193 CP3JB6 25181625 IC50 = 5.012 nM T83193 CPH98K 25181768 IC50 = 79 nM T83193 CG7HA8 25181770 IC50 = 23 nM T83193 CW9J5U 25181771 IC50 = 0.5012 nM T83193 CPZA63 25181773 IC50 = 0.631 nM T83193 CRAE91 25181908 IC50 = 43 nM T83193 C21MGD 25181909 IC50 = 46 nM T83193 CA78YZ 25181911 IC50 = 55 nM T83193 CT8SH5 25182164 IC50 = 87 nM T83193 CG2K6M 25182166 IC50 = 92 nM T83193 CG5K9X 25182169 IC50 = 392 nM T83193 CO73NW 25182447 IC50 = 0.631 nM T83193 CHR4D8 25182737 IC50 = 1.995 nM T83193 CVM90Z 25182893 IC50 = 12.59 nM T83193 CK7F2C 25195123 IC50 = 8.5 nM T83193 CRC21B 25241873 IC50 = 3.2 nM T83193 CI8SQ7 25263541 IC50 = 17 nM T83193 CTW7E8 25263542 IC50 = 150 nM T83193 C6DX5M 25264621 IC50 = 4 nM T83193 CJO5R6 25264622 IC50 = 16 nM T83193 C8AIY7 25264623 IC50 = 4 nM T83193 CE04YM 25264757 IC50 = 7 nM T83193 C32USM 25264907 IC50 = 6 nM T83193 CR4T9V 25264908 IC50 = 7 nM T83193 CJ50IN 25265057 IC50 = 6 nM T83193 C20XDK 25265635 IC50 = 40 nM T83193 C7FBO1 25270198 IC50 = 15 nM T83193 CL3KW6 25270199 IC50 = 4.8 nM T83193 C4U3OE 25840617 IC50 > 10000 nM T83193 C1B0ZO 25840619 IC50 > 10000 nM T83193 CBR69Y 25840620 IC50 > 10000 nM T83193 C1YN3E 27838559 IC50 = 1930 nM T83193 CS43UD 29372808 IC50 = 74 nM T83193 CS3U9T 30294430 IC50 = 59 nM T83193 C1YT6G 35368250 IC50 > 10000 nM T83193 CJX06W 36223059 Ki > 3000 nM T83193 CBR9U4 42613351 EC50 = 1000 nM T83193 C9QF7X 42617987 EC50 = 26400 nM T83193 CYB0L5 42617988 EC50 = 40 nM T83193 CJR92V 44189702 Ki = 0.49 nM T83193 C8S9PC 44271987 Ki = 1.46 nM T83193 C3IJC8 44271988 Ki = 1.4 nM T83193 C1FJV0 44272140 Ki = 0.71 nM T83193 CNLI07 44276258 Ki = 66.1 nM T83193 CF10YJ 44276297 Ki = 149 nM T83193 CCY37M 44334307 IC50 = 38 nM T83193 C2A1TY 44334308 Ki = 4 nM T83193 CHXW51 44334309 Ki = 11 nM T83193 CV6RC0 44334375 Ki = 330 nM T83193 CU4T5Q 44334391 IC50 = 2.4 nM T83193 CJ8U2P 44334401 Ki = 19 nM T83193 CP5M4B 44334439 Ki = 160 nM T83193 C63ZPI 44334455 Ki = 17 nM T83193 C07IZG 44334734 Ki = 1.4 nM T83193 C71XAD 44348204 EC50 = 5.012 nM T83193 CJ4BM2 44348288 EC50 = 199.53 nM T83193 CB6D5O 44348320 EC50 = 5.012 nM T83193 C6KMD9 44348328 EC50 = 19.95 nM T83193 CI5JL6 44348331 EC50 = 0.3981 nM T83193 C0LOT7 44366106 Ki = 4.6 nM T83193 C09VPI 44366285 Ki = 4 nM T83193 CV3W5G 44366327 Ki = 9.8 nM T83193 CR12UP 44366328 IC50 = 770 nM T83193 C3CKU0 44386779 IC50 = 0.4 nM T83193 C96REQ 44387739 IC50 > 10000 nM T83193 C8GYE2 44387747 IC50 = 526 nM T83193 C6GQB7 44387748 EC50 = 1160 nM T83193 C78BVO 44387749 IC50 = 1310 nM T83193 C3UQS8 44387754 EC50 = 618 nM T83193 CUP59X 44387767 IC50 = 12100 nM T83193 C5EIO1 44387768 EC50 = 5260 nM T83193 C17ZVR 44387769 IC50 = 334 nM T83193 C2Q6TB 44387771 IC50 = 2280 nM T83193 CIE4Q2 44387778 IC50 = 367 nM T83193 C7A3UJ 44387779 IC50 = 8130 nM T83193 C46CST 44387781 IC50 = 908 nM T83193 CFOH27 44391151 IC50 = 776 nM T83193 C8T6VB 44391169 IC50 = 3128 nM T83193 CG9D1C 44391183 IC50 = 2143 nM T83193 CL3QU4 44391189 IC50 = 726 nM T83193 C25KZQ 44391190 IC50 = 305 nM T83193 C6I0DX 44391210 IC50 = 948 nM T83193 CN90WE 44391216 IC50 = 10000 nM T83193 CU3XC1 44391232 IC50 = 5773 nM T83193 CW83NP 44391233 IC50 = 325 nM T83193 CC43MN 44391249 IC50 = 665 nM T83193 C7X3EZ 44391250 IC50 = 5447 nM T83193 C5R2SC 44395836 IC50 = 2796 nM T83193 CT84UQ 44395837 IC50 = 4867 nM T83193 CTY85S 44395850 IC50 > 10000 nM T83193 C9CO4K 44395916 IC50 = 2178 nM T83193 C0ZG1C 44395917 IC50 > 10000 nM T83193 C2Q3EG 44395921 IC50 > 10000 nM T83193 CCA71Z 44395934 IC50 > 10000 nM T83193 C76MTS 44395937 IC50 = 8.5 nM T83193 CG92UT 44395945 IC50 = 8590.7 nM T83193 C8CH9T 44395955 IC50 = 3825.8 nM T83193 CFU3Q9 44395965 IC50 > 10000 nM T83193 C05DPN 44395979 IC50 > 10000 nM T83193 CEV27Q 44395981 IC50 > 10000 nM T83193 CB67VI 44395992 IC50 = 279 nM T83193 C84DTU 44395995 IC50 > 10000 nM T83193 C2W4RX 44395996 IC50 > 10000 nM T83193 CON6R0 44396004 IC50 > 10000 nM T83193 CX9C2V 44396013 IC50 > 10000 nM T83193 C58JNY 44396021 IC50 > 10000 nM T83193 C31NUC 44396024 IC50 > 10000 nM T83193 CXCQ03 44396026 IC50 = 67.5 nM T83193 CJ1BR0 44396035 IC50 = 8118.8 nM T83193 C5HO1D 44396060 IC50 = 176.6 nM T83193 C8RP3K 44396061 IC50 = 1623 nM T83193 CNET70 44396064 IC50 = 2154 nM T83193 CFDE76 44396075 IC50 > 10000 nM T83193 C0GHL8 44396080 IC50 > 10000 nM T83193 CM8HA5 44396081 IC50 > 10000 nM T83193 CL91XU 44396083 IC50 = 57.7 nM T83193 CJPK65 44396086 IC50 > 25000 nM T83193 C3LFO6 44396088 IC50 > 10000 nM T83193 C7DN0E 44396089 IC50 > 10000 nM T83193 CY69FU 44396093 IC50 > 10000 nM T83193 COQE95 44396094 IC50 > 10000 nM T83193 CC4K5Q 44396107 IC50 > 10000 nM T83193 CJK3B7 44396111 IC50 > 10000 nM T83193 CCP3L4 44396112 IC50 = 340 nM T83193 C9F0TP 44396115 IC50 = 5745 nM T83193 CHKC63 44396118 IC50 > 10000 nM T83193 CVZ2R9 44396121 IC50 > 10000 nM T83193 CQX6S5 44396143 IC50 > 10000 nM T83193 C09WPE 44396145 IC50 = 300.7 nM T83193 CHD94P 44396146 IC50 = 893 nM T83193 CTD74U 44396150 IC50 = 5021 nM T83193 CXY71J 44396164 IC50 = 2727 nM T83193 CC52ZU 44396172 IC50 = 6169 nM T83193 C0JYQ8 44398602 IC50 = 2740 nM T83193 CCDT79 44398616 IC50 = 389.6 nM T83193 CZP60S 44398654 IC50 = 355.3 nM T83193 CJZB34 44398661 IC50 = 10380 nM T83193 C1U4DF 44398772 IC50 > 20000 nM T83193 CR47MA 44400841 IC50 = 1800 nM T83193 C8R1NG 44406816 IC50 = 49 nM T83193 CYS04D 44412342 IC50 = 470 nM T83193 CA87CB 44412350 IC50 = 640 nM T83193 C69TCS 44412351 IC50 = 22 nM T83193 CUV46O 44412359 IC50 = 224 nM T83193 CB6U8P 44412367 IC50 = 170 nM T83193 C8NU9I 44412368 IC50 = 320 nM T83193 CB6N0V 44412369 IC50 = 290 nM T83193 C0T8JU 44412401 IC50 = 24 nM T83193 CZ6EH0 44412449 IC50 = 340 nM T83193 CP29AX 44412456 IC50 = 1500 nM T83193 C2YW6P 44412457 IC50 = 160 nM T83193 CV92RL 44412465 IC50 = 2400 nM T83193 C0RT4W 44412466 IC50 = 1100 nM T83193 C81QGK 44416398 IC50 = 42 nM T83193 C6GX3K 44416399 IC50 = 233 nM T83193 C74DWR 44416414 IC50 = 3669 nM T83193 C1W3EM 44416415 IC50 = 387 nM T83193 CQ90TZ 44416416 IC50 > 4000 nM T83193 CF8I9J 44416417 IC50 = 624 nM T83193 CY7ZI6 44416441 IC50 = 1779 nM T83193 C0JM2B 44416470 IC50 = 91 nM T83193 CQW7G5 44416491 IC50 > 4000 nM T83193 CT2HX5 44416493 IC50 > 4000 nM T83193 CUK10L 44416494 IC50 > 4000 nM T83193 CG7W3F 44416519 IC50 = 60 nM T83193 C0T8MF 44416550 IC50 = 746 nM T83193 CUG3C2 44416551 IC50 > 4000 nM T83193 C6KJG8 44416573 IC50 = 1412 nM T83193 CV4SR3 44416597 IC50 = 4303 nM T83193 C3KN2W 44416619 IC50 = 1527 nM T83193 CS94LP 44416642 IC50 = 257 nM T83193 C6M8EL 44416643 IC50 = 131 nM T83193 CT1BK4 44416662 IC50 > 4000 nM T83193 CI0P3Q 44416754 IC50 = 974 nM T83193 C9MB0K 44416755 IC50 = 189 nM T83193 CHC7D3 44416759 IC50 > 4000 nM T83193 CP80IX 44416784 IC50 > 4000 nM T83193 CQ1A2Z 44416785 IC50 = 65 nM T83193 C9HA3I 44416788 IC50 > 4000 nM T83193 CR5U4E 44416860 IC50 > 4000 nM T83193 C8GLZ1 44416863 IC50 = 49 nM T83193 CXST24 44416878 IC50 = 417 nM T83193 CVN68O 44416879 IC50 = 24 nM T83193 CSB61J 44416900 IC50 = 377 nM T83193 C84IAM 44416931 IC50 = 158 nM T83193 CCA8J4 44416932 IC50 = 190 nM T83193 CLFO48 44416952 IC50 = 49 nM T83193 CCZ8G2 44416971 IC50 = 62 nM T83193 C32FIC 44416972 IC50 = 152 nM T83193 CZV6L3 44416973 IC50 = 39 nM T83193 C1UHR8 44417047 IC50 = 73 nM T83193 CPND83 44417048 IC50 > 4000 nM T83193 CF71AH 44417070 IC50 > 4000 nM T83193 C7RW0A 44417071 IC50 = 1502 nM T83193 CKM17E 44417074 IC50 = 91 nM T83193 CQE0Z5 44417075 IC50 = 168 nM T83193 C3JC2H 44426231 IC50 = 3750 nM T83193 C2HR7A 44426233 IC50 = 123 nM T83193 CRFB27 44430071 EC50 = 9.4 nM T83193 CY8JL9 44430072 EC50 = 4.6 nM T83193 CDTP25 44430073 EC50 = 25.5 nM T83193 CZHI60 44430074 EC50 = 4.7 nM T83193 C52AJN 44430075 EC50 = 51.5 nM T83193 C2CD1Z 44430076 EC50 = 69.5 nM T83193 CXC58F 44430077 EC50 = 1.9 nM T83193 C21OIG 44430078 EC50 = 15.2 nM T83193 C3JKY0 44430082 EC50 = 8.6 nM T83193 CX1TW8 44430086 EC50 = 7.9 nM T83193 CH9XY0 44433395 IC50 = 42 nM T83193 CFP90W 44444341 IC50 = 680 nM T83193 CI56CT 44444349 IC50 = 184 nM T83193 C7JF0C 44444350 Ki = 4 nM T83193 CIVW16 44444351 IC50 = 5 nM T83193 C0HL3F 44444357 IC50 = 19 nM T83193 CZ2KI3 44444374 Ki = 10 nM T83193 CO04XT 44444381 Ki = 22 nM T83193 C2BP8Z 44444392 Ki = 11 nM T83193 CZ03IW 44444394 Ki = 4 nM T83193 C5JX2M 44444395 Ki = 16 nM T83193 CWU59D 44444396 Ki = 2 nM T83193 CY64IB 44444397 IC50 > 1000 nM T83193 CSI8P9 44444398 Ki = 8 nM T83193 CM7X2P 44444399 Ki = 17 nM T83193 C8Z1RQ 44444400 Ki = 1 nM T83193 CWF8P0 44444401 Ki = 1 nM T83193 C0SM7N 44444918 IC50 = 11 nM T83193 CIF3H2 44447609 IC50 = 70 nM T83193 C8UMG2 44447610 IC50 = 14 nM T83193 CI67JP 44447611 IC50 = 790 nM T83193 C4H5ZI 44447612 IC50 = 1400 nM T83193 CC7J0M 44447613 IC50 > 10000 nM T83193 CXQ64G 44447614 IC50 = 220 nM T83193 CGV17K 44447615 IC50 > 10000 nM T83193 C98GNL 44447617 IC50 > 10000 nM T83193 C07OUB 44447618 IC50 = 253 nM T83193 CLX6H3 44447619 IC50 > 10000 nM T83193 CJI0F1 44447620 IC50 > 10000 nM T83193 C59OWX 44447621 IC50 > 10000 nM T83193 CE67YB 44447622 IC50 > 10000 nM T83193 C9IE0S 44447623 IC50 > 10000 nM T83193 CVXH28 44447624 IC50 = 6000 nM T83193 CPJ0I5 44447625 IC50 > 10000 nM T83193 CK0BR6 44447626 IC50 > 10000 nM T83193 C7TGS0 44447627 IC50 = 380 nM T83193 CN30TO 44447628 IC50 = 477 nM T83193 CLJ6B8 44447629 IC50 = 1420 nM T83193 C5VH4R 44447630 IC50 = 4970 nM T83193 C7IU4D 44447631 IC50 > 10000 nM T83193 CQ89RW 44447632 IC50 = 1310 nM T83193 C9JW1X 44447633 IC50 = 1640 nM T83193 CJ28NP 44447634 IC50 = 1730 nM T83193 CKTP16 44447635 IC50 = 3720 nM T83193 CJXI21 44447636 IC50 > 10000 nM T83193 C7S9OY 44447637 IC50 = 2620 nM T83193 CAF50B 44447638 IC50 = 205 nM T83193 CO4HF6 44447639 IC50 = 776 nM T83193 C5A1IB 44447641 IC50 = 2560 nM T83193 CCV8W3 44447642 IC50 = 3700 nM T83193 CA3TM9 44447648 IC50 = 1890 nM T83193 C7ZKH5 44447649 IC50 = 1160 nM T83193 C7AO1C 44447650 IC50 = 3430 nM T83193 C6J5TL 44447651 IC50 > 10000 nM T83193 COCQ06 44447652 IC50 > 10000 nM T83193 CK4OE2 44447653 IC50 = 3940 nM T83193 C1YR8I 44447654 IC50 = 3400 nM T83193 CPO9Q6 44447655 IC50 > 10000 nM T83193 C26JRZ 44447667 IC50 = 400 nM T83193 CHB65M 44447668 IC50 = 550 nM T83193 C7T2DQ 44447669 IC50 = 5070 nM T83193 C0Y7IX 44447670 IC50 = 3280 nM T83193 CYR56O 44447671 IC50 = 490 nM T83193 CL4HR0 44447672 IC50 = 200 nM T83193 CD80OW 44447673 IC50 = 2600 nM T83193 C0P1QK 44447674 IC50 > 10000 nM T83193 CC6M4A 44447675 IC50 = 6700 nM T83193 CN5W9K 44447676 IC50 = 4600 nM T83193 CW4PO2 44447677 IC50 = 5400 nM T83193 C0TY7X 44447678 IC50 = 7300 nM T83193 CWK61M 44447679 IC50 = 1400 nM T83193 CM6FB3 44447680 IC50 > 10000 nM T83193 C4YV8G 44447681 IC50 > 10000 nM T83193 CVL4W5 44447682 IC50 > 10000 nM T83193 CO5MJ1 44447683 IC50 = 4650 nM T83193 COW25J 44447684 IC50 = 3550 nM T83193 CRNM76 44447685 IC50 = 150 nM T83193 CHEP38 44447686 IC50 = 76 nM T83193 CSWN64 44447687 IC50 = 1230 nM T83193 CP3WU4 44447688 IC50 = 960 nM T83193 CFW8G9 44447689 IC50 = 1350 nM T83193 CF5EB0 44447690 IC50 = 3100 nM T83193 CAZ4E9 44447691 IC50 > 10000 nM T83193 CQB6I3 44447692 IC50 = 81 nM T83193 CHO2B5 44447693 IC50 = 740 nM T83193 CW1VH4 44447972 IC50 = 70 nM T83193 CIJB18 44447973 IC50 = 32 nM T83193 CRY47W 44448494 EC50 > 100000 nM T83193 CA49WS 44448505 EC50 > 100000 nM T83193 C6AY8U 44448506 EC50 = 29600 nM T83193 C7ZJ9O 44448536 EC50 > 100000 nM T83193 C72IYN 44448539 EC50 = 15000 nM T83193 CZTQ62 44448540 EC50 = 53500 nM T83193 C4G9YD 44448542 EC50 > 100000 nM T83193 CBA36L 44448576 EC50 > 100000 nM T83193 CSB9M8 44448577 EC50 > 100000 nM T83193 C0J4VA 44448578 EC50 > 100000 nM T83193 CGL3J5 44448579 EC50 > 100000 nM T83193 COWF13 44448613 EC50 > 100000 nM T83193 C7VGI3 44448615 EC50 > 100000 nM T83193 CIR53D 44448618 EC50 > 100000 nM T83193 CVB6E5 44448647 EC50 > 100000 nM T83193 CS9YA3 44448648 EC50 > 100000 nM T83193 C7JYR2 44448650 EC50 > 100000 nM T83193 C7FU4D 44450275 Ki = 16 nM T83193 CH76LB 44450299 Ki = 1471 nM T83193 C64CPA 44450314 Ki = 24 nM T83193 CEF47K 44450323 Ki = 38 nM T83193 CJC7Y0 44450337 IC50 > 30000 nM T83193 C5F1JL 44450338 Ki = 267 nM T83193 CU6Q2L 44450367 Ki > 3000 nM T83193 C52CIP 44450378 Ki > 3000 nM T83193 C67ZYA 44454325 IC50 = 10 nM T83193 C0LWU9 44454328 IC50 = 2.9 nM T83193 C6GZ8V 44454360 IC50 = 2.1 nM T83193 CC31AH 44566752 IC50 > 200000 nM T83193 CC9Q7V 44569302 IC50 = 539 nM T83193 C3VZY7 44569303 IC50 = 224 nM T83193 CBYE01 44569304 IC50 = 274 nM T83193 CY6O1V 44569360 IC50 = 5000 nM T83193 CO54EV 44569361 IC50 = 184 nM T83193 CSG9U4 44569441 IC50 = 59 nM T83193 CJ82AH 44569442 IC50 = 48 nM T83193 CX25DT 44569484 IC50 = 39 nM T83193 CTI30N 44569485 IC50 = 1 nM T83193 C9R5XV 44569566 IC50 > 5000 nM T83193 C8BN2K 44569567 IC50 = 680 nM T83193 C6N8YA 44569568 IC50 > 5000 nM T83193 C9TR7S 44569601 IC50 = 502 nM T83193 CVW69G 44569602 IC50 = 43 nM T83193 C03OFA 44569641 IC50 = 234 nM T83193 CJ2X4R 44569642 IC50 = 51 nM T83193 CC8WO2 44569643 IC50 = 74 nM T83193 CP9DQ2 44569644 IC50 > 5000 nM T83193 CLAV98 44569672 IC50 = 95 nM T83193 CRP64A 44569673 IC50 = 125 nM T83193 CGN01P 44569738 IC50 = 69 nM T83193 C5K7OD 44569739 IC50 = 820 nM T83193 CN5K2H 44569740 IC50 > 5000 nM T83193 CJT58N 44569741 IC50 > 5000 nM T83193 C3SU5I 44569781 IC50 > 5000 nM T83193 CNK24D 44569782 IC50 > 5000 nM T83193 CFZ3H1 44569783 IC50 = 206 nM T83193 CJH87Z 44569784 IC50 > 5000 nM T83193 COW7F2 44569785 IC50 = 176 nM T83193 CD4O8U 44569814 IC50 = 33 nM T83193 C5JAG6 44569815 IC50 = 10 nM T83193 C5YGU6 44569816 IC50 = 31 nM T83193 CA2W1E 44569847 IC50 = 96 nM T83193 C6Y1ZB 44569848 IC50 > 5000 nM T83193 CB9F4A 44569849 IC50 > 5000 nM T83193 CR6UV4 44569850 IC50 > 5000 nM T83193 CUQ39B 44569893 IC50 > 5000 nM T83193 CS89MB 44569894 IC50 = 1 nM T83193 CMJ97X 44570894 IC50 = 9.4 nM T83193 C9YTH7 44570896 IC50 = 32 nM T83193 C2IWK3 44570932 IC50 = 226 nM T83193 C15JVN 44570933 IC50 = 205 nM T83193 CS6D5L 44570976 IC50 = 80 nM T83193 C4OJ3F 44571024 IC50 = 81 nM T83193 CCE67G 44579757 IC50 = 67 nM T83193 CQ25HD 44579758 IC50 = 35 nM T83193 CZA30W 44579759 IC50 = 95 nM T83193 C78CWZ 44579760 IC50 = 196 nM T83193 C9P5KO 44580000 IC50 = 78 nM T83193 C2C7NM 44580001 IC50 = 27 nM T83193 CQ84AH 44580002 IC50 = 19 nM T83193 C15HBR 44580003 IC50 = 14 nM T83193 CO13LW 44580004 IC50 = 10 nM T83193 CV1O7Z 44580033 IC50 = 265 nM T83193 C64AFD 44580034 IC50 = 41 nM T83193 CQLO61 44585756 IC50 > 50000 nM T83193 CBT81W 44587581 IC50 = 46 nM T83193 C3OKQ1 44587671 IC50 = 81 nM T83193 CAG32Q 44587705 IC50 = 36 nM T83193 C0J5AB 44587803 IC50 = 890 nM T83193 C0F6IE 44587823 IC50 = 2 nM T83193 CF89OM 44587857 IC50 = 1 nM T83193 CM8YS9 44587934 IC50 = 2 nM T83193 CKRZ26 44755933 EC50 = 4800 nM T83193 C4WS8T 45375957 IC50 = 1000 nM T83193 C80GPZ 45380559 IC50 = 7 nM T83193 CLK8O9 45380748 IC50 = 32 nM T83193 C84ORB 45380848 IC50 = 5 nM T83193 CQDI48 46191427 IC50 = 10 nM T83193 CAT9Z8 46191428 IC50 = 5 nM T83193 CP08ZD 46191499 IC50 = 32 nM T83193 C0ET7O 46191501 IC50 = 5 nM T83193 C4HSX5 46191502 IC50 = 3 nM T83193 CSD13A 46191565 IC50 = 22 nM T83193 CXIC58 46191567 IC50 = 9 nM T83193 C71CGU 46191622 IC50 = 2 nM T83193 CUHT54 46202912 IC50 = 0.83 nM T83193 CBL4C0 46202914 IC50 = 0.21 nM T83193 C6RJ0G 46203233 IC50 = 665 nM T83193 CI6Y5Q 46203537 IC50 = 1.65 nM T83193 C0Q5CE 46203540 IC50 = 308 nM T83193 C97LXB 46203543 IC50 = 6.1 nM T83193 CMB32E 46203864 IC50 = 2.2 nM T83193 CYQG10 46203867 IC50 = 0.2 nM T83193 CCDL39 46203868 IC50 = 79 nM T83193 CS57CK 46204201 IC50 = 460 nM T83193 CGY31W 46225223 EC50 = 19 nM T83193 C3E0RS 46225224 EC50 = 17.4 nM T83193 CA08KQ 46225225 EC50 = 0.65 nM T83193 CECI47 46225226 EC50 = 0.98 nM T83193 C6DM4B 46225227 EC50 = 0.15 nM T83193 CQ31DN 46225228 EC50 = 13.7 nM T83193 C28VIE 46225229 EC50 = 0.0047 nM T83193 CP6Q0D 46847337 IC50 = 3.162 nM T83193 CK5DW1 46847339 IC50 = 3.981 nM T83193 C8XC1H 46862564 IC50 = 794.33 nM T83193 C0SJO4 46865592 IC50 = 79.43 nM T83193 CB70JQ 46865593 IC50 = 19.95 nM T83193 C7ICH3 46865714 IC50 = 5011.87 nM T83193 C7TVB4 46865715 IC50 = 1000 nM T83193 CLM61U 46865716 IC50 = 125.89 nM T83193 CBI2C3 46879825 IC50 = 480 nM T83193 CP4T7X 46879826 IC50 > 10000 nM T83193 CAQ5R4 46879827 IC50 > 10000 nM T83193 C3DZ7T 46879828 IC50 = 3900 nM T83193 CE35RZ 46879878 IC50 > 10000 nM T83193 CVI20B 46879879 IC50 > 10000 nM T83193 C7YUV0 46879880 IC50 > 10000 nM T83193 CQ7BG8 46879881 IC50 = 260 nM T83193 C17SUC 46879882 IC50 > 10000 nM T83193 C3KJD7 46879962 IC50 > 10000 nM T83193 CBK1A2 46879963 IC50 = 4600 nM T83193 C27SQX 46879964 IC50 > 10000 nM T83193 CVTM60 46879965 IC50 > 10000 nM T83193 C2TCG9 46880022 IC50 > 10000 nM T83193 CPH2B0 46880023 IC50 > 10000 nM T83193 C0DPM5 46880024 IC50 > 10000 nM T83193 CM79PR 46880025 IC50 > 10000 nM T83193 CQ8CZ3 46880026 IC50 > 10000 nM T83193 C2PQ6Z 46880080 IC50 > 10000 nM T83193 CA0S7Z 46880081 IC50 > 10000 nM T83193 C3F9BQ 46880082 IC50 > 10000 nM T83193 C6BUT5 46887685 EC50 = 250 nM T83193 CUR8T5 46887699 EC50 = 10 nM T83193 C2DSH4 46887729 EC50 = 7600 nM T83193 C37TUH 46887730 EC50 = 4100 nM T83193 CC4BM2 46887741 EC50 = 2.512 nM T83193 C3DNY1 46887742 EC50 = 6.31 nM T83193 C72YRJ 46887775 EC50 = 5800 nM T83193 CG5US0 46887776 EC50 = 18300 nM T83193 CDOZ92 46887777 EC50 = 7100 nM T83193 CEV8T0 46887779 EC50 = 19200 nM T83193 C3LTH4 46887780 EC50 = 42800 nM T83193 CC5VF3 46887829 EC50 = 53800 nM T83193 CF20RK 46887830 EC50 = 1000 nM T83193 CX13FH 46887831 EC50 = 52200 nM T83193 CR15JT 46887832 EC50 = 230 nM T83193 CA05CQ 46890470 IC50 = 3.5 nM T83193 C4ZQT8 46890471 IC50 = 16 nM T83193 C4S5NR 46890472 IC50 = 14 nM T83193 CW7M5V 46890473 IC50 = 12 nM T83193 CN9Q1V 46890474 IC50 = 125 nM T83193 CF2MP7 46890519 IC50 = 9 nM T83193 C0F1OT 46890520 IC50 = 18 nM T83193 CNZA79 46890521 IC50 = 12 nM T83193 CFE72M 46890522 IC50 = 6 nM T83193 CMY9Q7 46890558 IC50 = 5 nM T83193 CRJZ40 46890559 IC50 = 8 nM T83193 CZ5L4F 46890560 IC50 = 8 nM T83193 CK03BA 46890561 IC50 = 9 nM T83193 CFT95E 46890599 IC50 = 9 nM T83193 CERU86 46890600 IC50 = 6 nM T83193 CGY5O8 46890601 IC50 = 4.3 nM T83193 C3HM1E 46890636 IC50 = 53 nM T83193 C7OG8I 46890637 IC50 = 69 nM T83193 C4DTN2 46911175 IC50 = 0.8 nM T83193 CB71DC 47297796 IC50 > 1000 nM T83193 C4CG8H 49799019 IC50 = 864 nM T83193 C28LCD 49799119 IC50 = 840 nM T83193 C6ZES7 49799164 IC50 = 120 nM T83193 CEOA34 49799165 IC50 = 150 nM T83193 C8ZEV3 49799281 IC50 = 2.1 nM T83193 C5YB3J 49799282 IC50 = 114 nM T83193 CN4IA2 49799319 IC50 = 9 nM T83193 CL1Y3D 49799400 IC50 = 229 nM T83193 C0YX5G 49799401 IC50 = 101 nM T83193 CJ2O8F 49799402 IC50 = 10 nM T83193 C0PYK3 49799487 IC50 = 2 nM T83193 CIB0O2 49799488 IC50 = 1.3 nM T83193 CBI95M 49800487 Ki = 0.4 nM T83193 CJ9QN5 49800488 Ki = 31.7 nM T83193 C4A0WZ 49800489 Ki = 0.3 nM T83193 CG3YU6 49800490 Ki = 0.3 nM T83193 CBX1V7 49804209 Ki = 27.7 nM T83193 CQ73ET 49804501 Ki = 21.6 nM T83193 CPB17S 49804502 Ki = 0.3 nM T83193 C5ROS2 49804506 Ki = 8 nM T83193 CA2N7C 49804795 Ki = 75.2 nM T83193 C72LYO 49804796 Ki = 3.7 nM T83193 CU0R5J 49804798 Ki = 0.5 nM T83193 CXDY96 49863783 IC50 = 5.5 nM T83193 C04BIX 49863784 IC50 = 4.4 nM T83193 CN45OH 49863799 IC50 = 81 nM T83193 CCS97I 49863800 IC50 = 25.4 nM T83193 CTD96F 49863801 IC50 = 48.7 nM T83193 C61LAF 49863802 IC50 = 1450 nM T83193 CDC3E9 49863825 IC50 = 47 nM T83193 CO4CR7 49863826 IC50 = 161 nM T83193 C3YRI7 49863827 IC50 = 134 nM T83193 C79MBF 49863867 IC50 = 13 nM T83193 CG3R4U 49863868 IC50 = 607 nM T83193 CF1K6M 49863889 IC50 = 30 nM T83193 C91ZEV 49863890 IC50 = 15 nM T83193 CXP96N 49863891 IC50 = 27 nM T83193 CLWI96 49870854 IC50 = 11 nM T83193 C90UKY 50899643 IC50 > 10000 nM T83193 COTK61 52918271 IC50 = 1 nM T83193 CRU86C 52918272 IC50 = 2.512 nM T83193 C75OUP 52941151 IC50 = 2520 nM T83193 C9TIQ8 52941239 IC50 = 70 nM T83193 CI3Y7H 52941260 IC50 = 1450 nM T83193 C3CI1S 52941261 IC50 = 4220 nM T83193 CSHU46 52941328 IC50 > 20000 nM T83193 C7VU8Z 52941372 IC50 = 18 nM T83193 CBZ8P2 52941429 IC50 = 18 nM T83193 CR2DV9 52941523 IC50 = 56 nM T83193 CUN29Y 52942454 IC50 = 2780 nM T83193 C76CYL 52942485 IC50 = 1940 nM T83193 C86XKP 52942506 IC50 = 449 nM T83193 CZ7AR6 52942548 IC50 = 462 nM T83193 CEL6A4 52942660 IC50 = 51 nM T83193 CRO4D0 52942705 IC50 = 37 nM T83193 CT80GC 52943679 IC50 = 21 nM T83193 CE8Q9H 52943953 IC50 = 61 nM T83193 CIL01O 52943954 IC50 = 58 nM T83193 C68QPI 52944760 IC50 = 19 nM T83193 C6B5GL 52944788 IC50 = 25 nM T83193 C2ZVJ9 52944807 IC50 = 3350 nM T83193 CSYL32 52944808 IC50 = 52 nM T83193 C5IB7F 52944955 IC50 > 6670 nM T83193 CS05EZ 52944995 IC50 > 10000 nM T83193 C3R4BQ 52945186 IC50 = 230 nM T83193 C1R5QI 52945343 IC50 = 1058 nM T83193 CLZ2Y0 52945367 IC50 = 7.1 nM T83193 C8YG4L 52946049 IC50 = 43 nM T83193 C12TYW 52946120 IC50 = 2460 nM T83193 C9YUE3 52946246 IC50 = 56 nM T83193 CGPN15 52946286 IC50 = 31 nM T83193 C06ZDI 52946380 IC50 = 87 nM T83193 C6QD9F 52947296 IC50 = 2330 nM T83193 CI68FS 52947502 IC50 = 2040 nM T83193 CY25PM 52948674 IC50 = 176 nM T83193 C8CZE7 52949686 IC50 > 20000 nM T83193 C25JSC 52949800 IC50 = 520 nM T83193 CEK05T 52949901 IC50 = 580 nM T83193 CWBH28 52950142 IC50 = 180 nM T83193 CV53UF 53251173 IC50 = 718 nM T83193 CW7I3P 53251330 IC50 = 933 nM T83193 CS95ME 53257733 IC50 = 275000 nM T83193 CSXZ90 53259578 IC50 = 1665000 nM T83193 C8ZJ9V 53316531 IC50 = 3600 nM T83193 CAC4B1 53316588 IC50 = 367 nM T83193 C2M5DZ 53316589 IC50 = 41 nM T83193 CP5IX2 53316590 IC50 = 65 nM T83193 CWK47I 53317334 IC50 = 1380 nM T83193 CTM5Y0 53317849 IC50 = 1756 nM T83193 C68GBO 53318190 IC50 = 404 nM T83193 CIJ02V 53318736 IC50 = 15 nM T83193 CY48EJ 53318883 IC50 = 238 nM T83193 CFG6X9 53318884 IC50 = 197 nM T83193 CWQ51H 53319165 IC50 = 140 nM T83193 CQI0V6 53319221 IC50 = 132 nM T83193 CK7TX5 53319909 IC50 = 3330 nM T83193 C59MGC 53320201 IC50 = 762 nM T83193 C4DC2Y 53320280 IC50 = 115 nM T83193 C4MXJ2 53320373 IC50 > 5000 nM T83193 C9Z7JY 53320484 IC50 > 5000 nM T83193 CXE4K1 53320485 IC50 = 250 nM T83193 CXV68G 53320830 IC50 = 50.12 nM T83193 C8R2ZC 53320831 IC50 = 201 nM T83193 C67QBL 53321243 IC50 = 6 nM T83193 C1RDE5 53321779 IC50 = 498 nM T83193 C12JTH 53321780 IC50 = 2667 nM T83193 C9H5AL 53321781 IC50 = 3700 nM T83193 CT0QG8 53321782 IC50 = 62 nM T83193 CY0TR1 53321783 IC50 = 53 nM T83193 C01CMS 53321847 IC50 = 11 nM T83193 C30HUE 53322166 IC50 = 1252 nM T83193 CRJY79 53322568 IC50 = 853 nM T83193 C6IWP5 53322847 IC50 = 263 nM T83193 CTK26S 53322848 IC50 = 434 nM T83193 C5VGA6 53323109 IC50 = 2000 nM T83193 C9ZU3V 53323161 IC50 = 91 nM T83193 CP6TV2 53323958 IC50 = 1200 nM T83193 CTO91A 53324108 IC50 = 112 nM T83193 CK2D5S 53324459 IC50 = 100 nM T83193 CIP2R6 53324813 IC50 = 410 nM T83193 CIC87Z 53324814 IC50 = 112 nM T83193 CQL80G 53325473 IC50 = 149 nM T83193 C3GJ1P 53325573 IC50 = 377 nM T83193 C0MG2V 53325658 IC50 = 24 nM T83193 C86PXA 53325663 IC50 = 243 nM T83193 CWEF56 53325770 IC50 = 150 nM T83193 CH0SJ3 53325771 IC50 = 185 nM T83193 CHPB78 53325772 IC50 = 3080 nM T83193 CK2GH1 53325956 IC50 = 2790 nM T83193 C2S9QF 53326093 IC50 = 4222 nM T83193 C1ZB5W 53326094 IC50 = 370 nM T83193 CU71RE 53326526 IC50 = 31 nM T83193 CP8YN4 53326730 IC50 = 595 nM T83193 C3OU8Z 53326731 IC50 = 2212 nM T83193 COJ05G 53326732 IC50 = 120 nM T83193 CX4T7C 53326733 IC50 = 48 nM T83193 CQ1CA3 53326824 IC50 = 476 nM T83193 CHCV32 53326862 IC50 = 65 nM T83193 CN9XB7 53341424 IC50 = 2.8 nM T83193 CPD9E0 53341464 IC50 = 10 nM T83193 CCE3M7 53341467 IC50 = 22 nM T83193 C54RAO 53341468 IC50 = 7 nM T83193 CGM0P7 53341469 IC50 = 9.2 nM T83193 C1DEO5 53344884 IC50 = 2.8 nM T83193 C1PVA2 53363480 IC50 = 63.1 nM T83193 CSYK59 54580312 IC50 = 3.162 nM T83193 CDV60E 54580597 IC50 = 5.9 nM T83193 CC6MY2 54581318 IC50 = 25.12 nM T83193 CX4W9B 54581319 IC50 = 25.12 nM T83193 C2Z5MI 54581320 IC50 = 10 nM T83193 CD7T6A 54581321 IC50 = 7.943 nM T83193 C05UWK 54581568 IC50 = 87 nM T83193 CY96DR 54581578 IC50 = 6.1 nM T83193 CHK9X8 54581579 IC50 = 11 nM T83193 CH79VA 54581580 IC50 = 8 nM T83193 CI6DG4 54581581 IC50 = 12 nM T83193 CG5OY0 54581582 IC50 = 4.9 nM T83193 C7URO0 54581583 IC50 = 31 nM T83193 CH45CT 54581605 IC50 = 34 nM T83193 C8RBZ2 54581606 IC50 = 7.5 nM T83193 CRI4D6 54582331 IC50 = 15.85 nM T83193 C2QT8D 54582332 IC50 = 1258.93 nM T83193 CTLX27 54582573 IC50 > 1000 nM T83193 CBY8X7 54583542 IC50 = 14 nM T83193 CC62IP 54583543 IC50 = 1.7 nM T83193 CRXD15 54583544 IC50 > 1000 nM T83193 CU87MQ 54584525 IC50 = 52 nM T83193 CMKC41 54584526 IC50 = 24 nM T83193 COYG60 54584527 IC50 = 13 nM T83193 CM39GI 54584539 IC50 = 260 nM T83193 CL7P1G 54585233 IC50 = 7.943 nM T83193 CLH59Y 54585234 IC50 = 3162.28 nM T83193 CA3D6M 54585460 IC50 = 12 nM T83193 C9G7BI 54585461 IC50 = 7.5 nM T83193 CYSJ96 54585485 IC50 = 32 nM T83193 CS8GO5 54586192 IC50 = 0.1585 nM T83193 CJCT30 54586193 IC50 = 79.43 nM T83193 CVH34C 54586194 IC50 = 5.012 nM T83193 CJK4A9 54586430 IC50 = 28 nM T83193 CZ7UO6 54586431 IC50 > 1000 nM T83193 CB7OU9 54586432 IC50 = 520 nM T83193 CNZ87H 54586433 IC50 = 12 nM T83193 CF7N3X 54586458 IC50 = 44 nM T83193 CLAJ60 54587208 IC50 = 1.259 nM T83193 CHMU16 54587209 IC50 = 12.59 nM T83193 CXCT26 54587210 IC50 = 10 nM T83193 CY7WO8 54587294 IC50 = 1320000 nM T83193 CX6K9Z 54587295 IC50 = 227000 nM T83193 C1R8EC 54587460 IC50 = 5.7 nM T83193 CIY57J 54587479 IC50 = 340 nM T83193 CCO2I3 54587480 IC50 > 1000 nM T83193 C47PDY 54587481 IC50 = 6.8 nM T83193 CUV69N 54669855 EC50 = 4400 nM T83193 C2L3AP 56659764 IC50 = 199.53 nM T83193 CI51JF 56659769 IC50 = 125.89 nM T83193 CKY93J 56659770 IC50 = 158.49 nM T83193 CA13MO 56659771 IC50 = 5011.87 nM T83193 CIE1F0 56659772 IC50 = 316.23 nM T83193 CCBE24 56666677 IC50 = 158.49 nM T83193 C41IRL 56666678 IC50 = 794.33 nM T83193 CX3C4N 56670093 IC50 = 12.59 nM T83193 CCOP96 56670094 IC50 = 1584.89 nM T83193 CK9L6R 56673610 IC50 = 1584.89 nM T83193 COV8T6 56673613 IC50 = 1584.89 nM T83193 C64FYX 56676933 IC50 = 3162.28 nM T83193 CP0V8Y 56676934 IC50 = 1995.26 nM T83193 C57HIX 56676935 IC50 = 63.1 nM T83193 C2V7DN 56683573 IC50 = 3.162 nM T83193 C9WUS8 56683582 IC50 = 39.81 nM T83193 CRG8X7 56896484 IC50 = 314 nM T83193 C7TC2E 56966490 IC50 = 21 nM T83193 CY8NQ9 57334560 EC50 = 110 nM T83193 CDW28C 57334561 EC50 = 500 nM T83193 C34DKP 57334562 IC50 > 10000 nM T83193 C8OTV0 57334563 IC50 > 10000 nM T83193 C96KIT 57334564 IC50 > 50000 nM T83193 CADV61 57390833 IC50 > 100000 nM T83193 CH6D3G 57392653 IC50 > 50000 nM T83193 C6J5IZ 57394365 IC50 > 50000 nM T83193 CWD30P 57394366 IC50 > 10000 nM T83193 C19LBS 57394367 EC50 = 100 nM T83193 CIX28C 57396122 EC50 = 14600 nM T83193 CZ9DL6 57397938 IC50 > 50000 nM T83193 C5MU1H 57397939 EC50 = 14300 nM T83193 CIXP67 57399580 IC50 = 35300 nM T83193 CQ5P7U 57401337 IC50 = 4800 nM T83193 C32NVG 57927125 IC50 = 320 nM T83193 CL10GR 58381102 IC50 = 6 nM T83193 CQV67K 58381208 IC50 = 19 nM T83193 CVY71G 58543815 IC50 > 100000 nM T83193 C0AI3H 58639564 IC50 = 750 nM T83193 C19NCQ 58755739 Ki = 217 nM T83193 CIV21U 58873250 Ki = 2.5 nM T83193 C1QJN0 58873252 Ki = 0.7 nM T83193 C42NXZ 58873256 Ki = 8.7 nM T83193 CL8IE5 58873257 Ki = 142 nM T83193 C9NU8M 58873260 Ki = 4 nM T83193 C5API8 58873263 Ki = 2 nM T83193 C7L2MN 58873266 Ki = 2.1 nM T83193 CQFL38 58873268 Ki = 0.7 nM T83193 C3V9HU 58873274 Ki = 0.3 nM T83193 C37AKC 58873277 Ki = 0.9 nM T83193 CKJ8B5 58873278 Ki = 14.6 nM T83193 CY47JC 58873281 Ki = 1.43 nM T83193 CMC0K2 58873283 Ki = 2.8 nM T83193 C61IXR 58873285 Ki = 2.9 nM T83193 CN4AE9 58873286 Ki = 1.8 nM T83193 C20NLZ 58873288 Ki = 0.7 nM T83193 C6UT7V 58873299 Ki = 1 nM T83193 CCI49K 58873310 Ki = 0.6 nM T83193 CME01F 58873315 Ki = 0.9 nM T83193 C92XOC 58873319 Ki = 0.6 nM T83193 CJUG90 58873320 Ki = 36.1 nM T83193 CFG70L 58873323 Ki = 146 nM T83193 C5WQ2C 58873326 Ki = 2.9 nM T83193 C63DYW 58873336 Ki = 1.2 nM T83193 CBZU20 58873340 Ki = 1.8 nM T83193 CP9Q3K 58873345 Ki = 7.7 nM T83193 CM3RC0 58873352 Ki = 1.3 nM T83193 CL74KX 58873360 Ki = 25.6 nM T83193 C2LF0B 58873361 Ki = 0.4 nM T83193 CFRO67 58873367 Ki = 0.8 nM T83193 CDO01G 58873371 Ki = 0.7 nM T83193 CB9TN3 58873374 Ki = 3.4 nM T83193 CG37QC 58873376 Ki = 13.8 nM T83193 C9NB8V 58873379 Ki = 0.8 nM T83193 CH21ET 58873383 Ki = 0.8 nM T83193 CEV28U 58873386 Ki < 1000 nM T83193 C14SMQ 58873396 Ki = 20.4 nM T83193 CNHX52 58873403 Ki = 3.2 nM T83193 CBK28Y 58873408 Ki = 4.2 nM T83193 C8YAB1 58873411 Ki = 2.3 nM T83193 CWT26G 58873412 Ki = 0.9 nM T83193 CU81DX 58873414 Ki = 0.8 nM T83193 CEN4Y5 58873424 Ki = 5.8 nM T83193 CTS30F 58873427 Ki = 0.3 nM T83193 CFL8W2 58873438 Ki = 15.3 nM T83193 C1FC4S 58873447 Ki = 1.9 nM T83193 CO47KG 58873448 Ki = 1.3 nM T83193 C9M2QG 58873450 Ki = 0.5 nM T83193 CWP8X0 58873451 Ki = 2.5 nM T83193 CRZS39 58873454 Ki = 0.7 nM T83193 C1UV7I 58873461 Ki = 51 nM T83193 C39AWE 58873465 Ki = 8.6 nM T83193 CLT9Z1 58873467 Ki = 2.5 nM T83193 CNET76 58873468 Ki = 2.5 nM T83193 CEN23Q 58873470 Ki = 1.7 nM T83193 C3VFN0 58873473 Ki = 0.7 nM T83193 CR8YK9 58873474 Ki = 2.7 nM T83193 CQ6SE3 58873475 Ki = 0.7 nM T83193 CDZ35O 58873481 Ki = 0.7 nM T83193 CG4NB0 58873497 Ki = 0.8 nM T83193 CCO6D0 58873499 Ki = 1.6 nM T83193 C61YMS 58873504 Ki = 3.2 nM T83193 C6GZT3 58873505 Ki = 0.6 nM T83193 CNKA45 58873506 Ki = 0.8 nM T83193 C6Q7FU 58873513 Ki = 65.7 nM T83193 CWI9U6 58873514 Ki = 1 nM T83193 CV3OU4 58873516 Ki = 0.4 nM T83193 C6IX7N 58873517 Ki = 68.7 nM T83193 C9EPG7 58873529 Ki = 1.9 nM T83193 C02TSG 58873530 Ki = 4.4 nM T83193 CQB4G1 58873536 Ki = 4.4 nM T83193 CDNF58 58873545 Ki = 91 nM T83193 C41BJQ 58873549 Ki = 39.3 nM T83193 CYJ73G 58873550 Ki = 0.001 nM T83193 C9T0NB 58873556 Ki = 0.5 nM T83193 CE4BO0 58873559 Ki = 3 nM T83193 CF7PH2 58873561 Ki = 0.5 nM T83193 CPK9D3 58873562 Ki = 43.7 nM T83193 CTJX93 58873563 Ki = 0.7 nM T83193 CWZ91P 58873575 Ki = 2.4 nM T83193 C1Y6GE 58873578 Ki = 2.2 nM T83193 CLBE06 58873579 Ki = 1 nM T83193 C3JP5E 58873581 Ki = 0.04 nM T83193 CW36FK 58873584 Ki = 1.5 nM T83193 CCI1S0 58873592 Ki = 1.5 nM T83193 C7B0FK 58873593 Ki = 2.5 nM T83193 C5OJI2 58873598 Ki = 8.1 nM T83193 C8D0XQ 58873600 Ki = 12.7 nM T83193 CU9SY5 58873608 Ki = 29.5 nM T83193 CY9FU3 58873610 Ki = 0.3 nM T83193 CG18HW 58873616 Ki = 1.6 nM T83193 C6J9MV 58873625 Ki = 44 nM T83193 CR4XA7 58873626 Ki = 15.8 nM T83193 CCB69W 58873638 Ki = 6.4 nM T83193 CUW53L 58873640 Ki = 1.1 nM T83193 C8C7MW 58873642 Ki = 0.5 nM T83193 C50PHI 58873652 Ki = 0.9 nM T83193 C3MB6C 58873654 Ki = 0.2 nM T83193 CJ72CP 58873655 Ki = 1 nM T83193 CY1HG9 58873658 Ki = 0.9 nM T83193 CI0MC5 58873667 Ki = 0.6 nM T83193 C7ZN6P 58873674 Ki = 16 nM T83193 C8K1XH 58873675 Ki = 4.4 nM T83193 CCXH69 58873678 Ki = 0.9 nM T83193 CDG2Z6 58873681 Ki = 0.9 nM T83193 CJDS23 58873682 Ki = 0.5 nM T83193 C7HR9E 58873691 Ki = 63.3 nM T83193 CQ2VK5 58873692 Ki = 2.7 nM T83193 C82NCS 58873694 Ki = 0.6 nM T83193 CG09QP 58873697 Ki = 9.7 nM T83193 CYD4M9 58873698 Ki = 0.3 nM T83193 CEI47W 58873712 Ki = 1.6 nM T83193 C7JOV4 58873713 Ki = 59.6 nM T83193 C5SNQ0 58873716 Ki = 0.7 nM T83193 C1CN7E 58873717 Ki = 1.6 nM T83193 CSHP94 58873734 Ki = 1.6 nM T83193 CIZN23 58873735 Ki = 3.3 nM T83193 CW4XP9 58873742 Ki = 17.5 nM T83193 CAY81O 58873745 Ki = 0.4 nM T83193 CPK63B 58873748 Ki = 1 nM T83193 C2QH3P 58873756 Ki = 0.7 nM T83193 CKJ40C 58873760 Ki = 0.8 nM T83193 CA13EB 58873763 Ki = 1 nM T83193 C48FVB 58873765 Ki = 0.8 nM T83193 CVC98P 58873771 Ki = 4.8 nM T83193 C91BTK 58873774 Ki = 2.4 nM T83193 CE36NO 58873778 Ki = 2.8 nM T83193 CB98IU 58873784 Ki = 19.3 nM T83193 CC63GV 58873793 Ki = 1.8 nM T83193 C9KNA0 58873796 Ki = 2.1 nM T83193 C3E9RN 58873810 Ki = 1.4 nM T83193 CH64QG 59007833 IC50 = 8 nM T83193 C7YT8V 59007841 IC50 = 22 nM T83193 CQ03ID 59007872 IC50 = 7 nM T83193 C6HDS2 59007884 IC50 = 240 nM T83193 CH6NX5 59007900 IC50 = 7 nM T83193 CSZ0B9 59007942 IC50 = 20 nM T83193 CSL09Q 59007969 IC50 = 5.9 nM T83193 C6J2ML 59008004 IC50 = 190 nM T83193 C0GFE3 59008008 IC50 = 17 nM T83193 CQ76CT 59008012 IC50 = 26 nM T83193 C4I1ME 59008027 IC50 = 13 nM T83193 CAM28G 59008035 IC50 = 40 nM T83193 C72EBR 59008085 IC50 = 4.5 nM T83193 CK79PR 59666268 IC50 = 93 nM T83193 C06TKS 59666298 IC50 = 87 nM T83193 CUN39P 60011733 IC50 = 180 nM T83193 C3VZ4T 60021981 IC50 = 16 nM T83193 C1Z0PC 60022072 IC50 = 56 nM T83193 CUH87T 66644289 Ki = 26.5 nM T83193 CM79IJ 67438722 Ki = 1.1 nM T83193 CTH71U 67438734 Ki = 1.3 nM T83193 C3CHO9 67439038 Ki = 2.3 nM T83193 CRS75Y 67439048 Ki = 100 nM T83193 CM02ZH 67439190 Ki = 3.7 nM T83193 CABX60 67439400 Ki = 14.8 nM T83193 CZ82FC 67439430 Ki = 2.1 nM T83193 C98OFW 67439460 Ki = 0.8 nM T83193 C0MUZ3 67439540 Ki = 3 nM T83193 CO0QB2 67439554 Ki = 1.4 nM T83193 CW4I6M 67439763 Ki = 0.4 nM T83193 CH1NR3 67439768 Ki = 3.4 nM T83193 CY70SV 67439821 Ki < 1000 nM T83193 C4VW6Q 67439823 Ki = 3.8 nM T83193 C32ONF 67439992 Ki = 5.6 nM T83193 CXF3U6 67440023 Ki = 0.7 nM T83193 CY79ZC 67440125 Ki = 0.9 nM T83193 CR2K7S 67440200 Ki = 4.2 nM T83193 CA03ES 67440314 Ki = 14.3 nM T83193 C1Y3QE 67440351 Ki = 2.1 nM T83193 C10CJQ 67440400 Ki = 0.8 nM T83193 CGB6I3 67440621 Ki = 2.2 nM T83193 CW8CK3 67440652 Ki = 1.7 nM T83193 C23SYL 67440783 Ki = 11.5 nM T83193 C1FK5L 67440786 Ki = 0.7 nM T83193 C38NTG 67440919 Ki = 0.4 nM T83193 C6AF8R 67440951 Ki = 5 nM T83193 CW07HE 67441243 Ki = 0.7 nM T83193 CV8T9K 67441528 Ki = 4.1 nM T83193 C63IOB 67441550 Ki = 20.3 nM T83193 CJM17W 67441632 Ki = 0.8 nM T83193 CX5PT0 67441643 Ki = 4 nM T83193 CM92GF 67441906 Ki = 23.9 nM T83193 C49ZSB 68653853 Ki = 22.7 nM T83193 C8DBE3 68718852 Ki = 48.7 nM T83193 C04EJH 68718961 Ki = 31.1 nM T83193 CBSY42 68721207 Ki = 37.6 nM T83193 C5OXZ3 69830044 IC50 > 1000 nM T83193 C4T1EY 69830874 IC50 = 34 nM T83193 C6D9XF 69903675 IC50 = 530 nM T83193 C1I6GO 70681468 IC50 = 230 nM T83193 C3T8HN 70682776 IC50 > 10000 nM T83193 CA0FG3 70682777 IC50 > 10000 nM T83193 C3ZKG0 70683578 IC50 = 45 nM T83193 CE6T5P 70683579 IC50 = 140 nM T83193 CNK40G 70684861 IC50 > 10000 nM T83193 CFDV81 70684862 IC50 = 833 nM T83193 CABQ74 70685686 IC50 = 9.1 nM T83193 CX3L9A 70685687 IC50 > 1000 nM T83193 CL0IK9 70685694 IC50 = 220 nM T83193 C4OFS1 70685695 IC50 = 330 nM T83193 CDJ51K 70687840 IC50 = 18 nM T83193 CFS60E 70687841 IC50 = 710 nM T83193 CN9B7M 70689871 IC50 = 130 nM T83193 C91TQS 70689872 IC50 > 1000 nM T83193 C1MLN9 70689873 IC50 = 460 nM T83193 CKX5D0 70692033 IC50 = 84 nM T83193 C25FYO 70694071 IC50 = 30 nM T83193 CMJ68Z 70694078 IC50 > 1000 nM T83193 CM70ZK 70898363 EC50 = 4897.79 nM T83193 CD6BV5 71237020 Ki = 8.4 nM T83193 C36KJR 71237040 Ki = 0.7 nM T83193 CI5NQ7 71237069 Ki = 7.1 nM T83193 C8M9YX 71237098 Ki = 0.4 nM T83193 C8FH5A 71237137 Ki = 1.8 nM T83193 C7XMW4 71237161 Ki = 8.9 nM T83193 CU52OL 71237192 Ki = 7.2 nM T83193 CI18GC 71237213 Ki = 9.5 nM T83193 CANF28 71237326 Ki = 0.02 nM T83193 CYU80Z 71237407 Ki = 91.6 nM T83193 C5U7AF 71237443 Ki = 48.1 nM T83193 CFHJ43 71237649 Ki = 7.8 nM T83193 CM9P0Z 71449757 IC50 = 1995.26 nM T83193 CSDE19 71449975 Ki = 0.2 nM T83193 CW3J4K 71450023 Ki = 0.3 nM T83193 C1BZR6 71451555 IC50 = 3162.28 nM T83193 C4X5RC 71451556 IC50 = 7943.28 nM T83193 CE45PR 71453396 IC50 = 1258.93 nM T83193 C5SEQ9 71453410 IC50 = 1584.89 nM T83193 CPA80H 71453411 IC50 = 630.96 nM T83193 C39LVF 71453662 Ki = 0.2 nM T83193 CWS2T3 71453663 Ki = 1.4 nM T83193 C27XOP 71455090 IC50 = 5011.87 nM T83193 C4JH2D 71455346 Ki = 11 nM T83193 CL86AH 71455347 Ki = 0.3 nM T83193 C2PL5G 71456898 IC50 = 794.33 nM T83193 CE2M1B 71456899 IC50 = 100 nM T83193 CUEX93 71456916 IC50 = 158.49 nM T83193 C6QVT0 71456917 IC50 = 1000 nM T83193 C3M9KC 71456918 IC50 = 501.19 nM T83193 CCF78E 71456919 IC50 = 3981.07 nM T83193 C6COI9 71457119 Ki = 0.4 nM T83193 CK28DR 71457120 Ki = 3.9 nM T83193 C6VU3T 71457121 Ki = 0.01 nM T83193 CE27CB 71457122 Ki = 7.5 nM T83193 CLDG16 71457160 Ki = 101 nM T83193 CPV3O2 71458753 IC50 = 1000 nM T83193 CM2F1A 71458754 IC50 = 2511.89 nM T83193 CPST04 71458774 IC50 = 1258.93 nM T83193 CZX76C 71458990 Ki = 2.1 nM T83193 C6NK2W 71458991 Ki = 9.8 nM T83193 CPQ4C6 71459032 Ki = 103 nM T83193 C0JB7W 71460583 IC50 = 199.53 nM T83193 CN0TC6 71460584 IC50 = 501.19 nM T83193 C1IKD0 71460788 Ki = 7.1 nM T83193 CKW28L 71460827 Ki = 2.6 nM T83193 CKP7J0 71462280 IC50 = 5011.87 nM T83193 CKO8C9 71462281 IC50 = 501.19 nM T83193 CKYO86 71462283 IC50 = 251.19 nM T83193 CX4OP7 71462545 Ki = 27.2 nM T83193 C4W8XS 71517050 IC50 = 440 nM T83193 C28CKU 71517051 EC50 = 6420 nM T83193 C1RG2N 71517052 EC50 = 11800 nM T83193 C0B2JQ 71517053 EC50 = 5100 nM T83193 C2HK8W 71517054 IC50 = 6400 nM T83193 C7T0YV 71517055 IC50 = 5100 nM T83193 C86OEX 71517056 EC50 = 400 nM T83193 C0ZGK9 71517199 EC50 = 5200 nM T83193 CE2UH4 71517200 EC50 = 7750 nM T83193 CDQ20R 71517201 EC50 = 1890 nM T83193 C5WE8T 71517202 IC50 = 1 nM T83193 CTL61C 71517203 EC50 = 7430 nM T83193 CQTR79 71517204 EC50 = 260 nM T83193 CG7FR3 71517205 EC50 = 2270 nM T83193 C7YH9K 71517356 EC50 = 170 nM T83193 C64RHP 71517357 EC50 = 1200 nM T83193 CX8HQ4 71517358 EC50 = 470 nM T83193 C6S8HN 71517359 EC50 = 5290 nM T83193 CD41WT 71517360 EC50 = 2400 nM T83193 C9O4FN 71517361 IC50 = 4360 nM T83193 CS46UC 71519502 IC50 = 9300 nM T83193 CQ0N9J 71519503 IC50 = 10600 nM T83193 CRK85C 71519504 IC50 = 9600 nM T83193 CM67KB 71528847 EC50 = 18620.87 nM T83193 CICU74 71537378 Ki = 6.77 nM T83193 C9HJ6P 71538504 Ki = 27.6 nM T83193 CT8OU5 71625073 IC50 = 516 nM T83193 CR0NS1 71625201 IC50 = 583 nM T83193 C1YG3H 71625202 IC50 = 33 nM T83193 CF4D3Z 71625203 IC50 = 130 nM T83193 C57ABI 71625204 IC50 = 44 nM T83193 CDG3B5 71625205 IC50 = 2620 nM T83193 CB7R9O 71625206 IC50 = 796 nM T83193 CGH9Q3 71625318 IC50 > 10000 nM T83193 C4F5XT 71625319 IC50 = 110 nM T83193 CQ31CB 71625320 IC50 > 10000 nM T83193 CB6Z0H 71625321 IC50 > 10000 nM T83193 C4F7LM 71625322 IC50 = 107 nM T83193 CXZ51P 71625323 IC50 = 86 nM T83193 CIMO89 71625324 IC50 = 941 nM T83193 CP74ZA 71698456 Ki = 1.3 nM T83193 C4JI2R 71698540 Ki = 0.3 nM T83193 C7NFG8 71698721 Ki = 0.3 nM T83193 CE6BS4 71698888 Ki = 2.6 nM T83193 C34HYQ 71698889 Ki = 0.8 nM T83193 CNE29A 71698890 Ki = 4.9 nM T83193 CXT35W 71698979 Ki = 1 nM T83193 CHRY76 71698980 Ki = 2.6 nM T83193 C0GJ2K 71699635 Ki = 49 nM T83193 CBT0I6 71699636 Ki = 50 nM T83193 CFTM13 71812230 EC50 = 0.99 nM T83193 CW20HQ 71818431 IC50 = 1260 nM T83193 C2L7TX 71818575 IC50 = 6300 nM T83193 C4IP1G 72197089 EC50 = 5900 nM T83193 C9EVP5 72197090 EC50 = 13400 nM T83193 CUAX51 72197091 EC50 = 1500 nM T83193 CWP34U 72197092 EC50 = 2500 nM T83193 CDN29K 72197093 EC50 = 1800 nM T83193 CA9CX5 72197094 EC50 = 250 nM T83193 C5QGC9 72197264 EC50 = 1700 nM T83193 C3C5FR 72197265 EC50 = 11900 nM T83193 CO5Z4D 72197266 IC50 > 100000 nM T83193 CX1J5H 72197267 IC50 > 100000 nM T83193 CXS6H8 72197268 IC50 > 100000 nM T83193 COMJ27 72197269 IC50 > 100000 nM T83193 CC95RF 72197270 IC50 > 100000 nM T83193 CSB3M1 72197441 EC50 = 25000 nM T83193 CC26EQ 72197442 IC50 > 100000 nM T83193 C2HD9F 72197443 EC50 = 32300 nM T83193 CV9DU7 72197444 IC50 > 100000 nM T83193 C9F1KH 72197445 IC50 > 100000 nM T83193 C0KL4H 72197446 EC50 = 22500 nM T83193 CO9TL8 72197447 IC50 > 100000 nM T83193 CHF0K8 72197628 IC50 > 100000 nM T83193 C5UT4O 72197629 IC50 > 100000 nM T83193 CNB9D0 72197630 IC50 > 100000 nM T83193 CT8LB2 72197631 IC50 > 100000 nM T83193 COJ5V6 72197632 IC50 > 100000 nM T83193 CVB7R8 72197633 IC50 > 100000 nM T83193 CVUH81 72197634 IC50 = 91800 nM T83193 C6W2NK 72197807 IC50 > 100000 nM T83193 C9VGP6 72197808 IC50 = 78900 nM T83193 C1Q5DT 72197809 EC50 = 4800 nM T83193 C28SBK 72203625 Ki = 2.3 nM T83193 CFP71H 72203627 Ki = 27.4 nM T83193 C2E3CW 72203628 Ki = 3.3 nM T83193 CH47JO 72203629 Ki = 3 nM T83193 CAG12S 72203823 Ki = 2.9 nM T83193 CT5OI8 72203826 Ki = 48.2 nM T83193 C8NK7U 72203827 Ki = 85 nM T83193 CV8Y0S 72204004 Ki = 1.2 nM T83193 CI1Q5C 72204007 Ki = 0.5 nM T83193 C16QGV 72204008 Ki = 1.9 nM T83193 CSG97M 72204177 Ki = 1 nM T83193 CTS3X9 72204178 Ki = 2.6 nM T83193 C7J0UX 72204179 Ki = 2.3 nM T83193 CM70LI 72204180 Ki = 8.7 nM T83193 CKF0D1 72204181 Ki = 3.2 nM T83193 C65HFT 72204376 Ki = 2.3 nM T83193 C9E6WU 72204377 Ki = 4.9 nM T83193 CZFU81 72204378 Ki = 3.9 nM T83193 CX7H6K 72204379 Ki = 14.6 nM T83193 CT81FE 72204380 Ki = 15 nM T83193 CUL51P 72204570 Ki = 1.9 nM T83193 CD1HF7 72204571 Ki = 0.05 nM T83193 CA1D0M 72204572 Ki = 43.5 nM T83193 C96BEP 72205499 IC50 = 841.6 nM T83193 CXR7L8 72205500 IC50 > 1000 nM T83193 CO57MJ 72205501 IC50 > 1000 nM T83193 C74JTD 72205502 IC50 = 266.3 nM T83193 C8NT4P 72205682 IC50 = 217.8 nM T83193 CDI82J 72205683 IC50 = 412.9 nM T83193 C16WFJ 72206428 Ki = 2.5 nM T83193 C34URG 72206429 Ki = 5.6 nM T83193 C1LP7R 72206430 Ki = 0.7 nM T83193 C2FL5C 72206431 Ki = 4.3 nM T83193 CN48VY 72206432 Ki = 7 nM T83193 CM13IT 72946681 Ki = 6.58 nM T83193 C5LP9N 72946682 Ki = 17.2 nM T83193 C5AQ2V 72946683 Ki = 63 nM T83193 C01WJG 73347328 IC50 = 411 nM T83193 CZ7U6Y 73349242 Ki = 330 nM T83193 COH89Q 73350826 EC50 = 16.5 nM T83193 CZB6C3 73352314 Ki = 212 nM T83193 CBDT72 73353428 Ki = 0.5 nM T83193 CDW07U 73355312 EC50 = 16.3 nM T83193 CW6ZP3 73355313 Ki = 50 nM T83193 CJQL93 73355314 Ki = 33.3 nM T83193 CEN85W 73355315 EC50 = 6.28 nM T83193 CC56EI 73356500 Ki = 1.5 nM T83193 C7QG1L 73356858 Ki = 990 nM T83193 CMF59G 73356859 EC50 = 17.9 nM T83193 CYT0M3 76327921 IC50 = 34 nM T83193 CR62OL 76335194 IC50 = 97 nM T83193 CXJI74 87401321 Ki = 0.9 nM T83193 CD9TA0 89469070 Ki = 199 nM T83193 CW12XC 89717400 IC50 = 70000 nM T83193 CXUH46 90645310 IC50 > 10000 nM T83193 CL0O7Q 90645312 IC50 > 10000 nM T83193 CN61RW 90645447 IC50 > 30000 nM T83193 CISP03 90645459 IC50 = 16700 nM T83193 CM5FN9 90645460 IC50 = 5100 nM T83193 C31TXQ 90645465 IC50 > 30000 nM T83193 C6OF3B 90645468 IC50 = 8100 nM T83193 C0VW1K 90645470 IC50 = 11500 nM T83193 C6SU4X 90665452 IC50 > 3900 nM T83193 CJCR26 90665456 IC50 > 16000 nM T83193 C7Y3DA 92045037 Ki = 1.99 nM T83193 COGJ67 92131136 Ki = 0.03 nM T83193 CF1D6S 101898797 EC50 = 6900 nM T83193 CVZ14O 101922675 EC50 = 2600 nM T83193 CFYD15 110877153 IC50 = 6100 nM T83193 CDNC39 118246723 IC50 > 30000 nM T83193 CEJ1A3 118707572 Ki = 22.7 nM T83193 CYC47B 118707573 Ki = 0.3 nM T83193 CQH41Y 118707574 Ki = 0.4 nM T83193 CK10OS 118707575 Ki = 0.3 nM T83193 CL6VZ5 118707576 Ki = 0.2 nM T83193 CPS2D8 118707577 Ki = 0.3 nM T83193 C9O3FI 118707578 Ki = 0.4 nM T83193 C75WKY 118707579 Ki = 0.3 nM T83193 C3C5NE 118707580 Ki = 1.5 nM T83193 CES2D3 118707581 Ki = 1.5 nM T83193 C7Q8GM 118707582 Ki = 0.8 nM T83193 CP3Y7C 118707583 Ki = 0.3 nM T83193 CQ17KB 118707584 Ki = 0.2 nM T83193 C0CIH4 118707585 Ki = 0.2 nM T83193 C21JUV 118707586 Ki = 0.1 nM T83193 CMAR-86 118707587 Ki = 0.1 nM T83193 CDBN38 118707588 Ki = 0.2 nM T83193 C8CIT6 118707589 Ki = 0.1 nM T83193 CE1B7V 118707590 Ki = 0.2 nM T83193 CQ4ZN2 118707591 Ki = 0.1 nM T83193 C3R5OM 118708168 Ki = 2 nM T83193 CQN36C 118708169 Ki = 5.8 nM T83193 CFX49V 118708170 Ki = 1.4 nM T83193 C9J1NK 118708171 Ki = 1 nM T83193 CO9EJ8 118708172 Ki = 141 nM T83193 CZH02O 118711168 IC50 > 200000 nM T83193 CT91SV 118711722 IC50 = 5 nM T83193 CO60KW 118711975 IC50 = 74 nM T83193 C1P0DX 118711976 IC50 = 97 nM T83193 C1X9PL 118711977 IC50 = 60 nM T83193 C9AGF7 118711978 IC50 = 350 nM T83193 C0A5NJ 118711979 IC50 = 22 nM T83193 CH1Q9Y 118711980 IC50 = 36 nM T83193 CP7N2U 118720705 EC50 = 6000 nM T83193 CFL2M7 118720706 IC50 > 100000 nM T83193 C29ZPL 118720707 IC50 > 100000 nM T83193 CUP7E9 118720708 IC50 > 100000 nM T83193 CPBE74 118720709 IC50 > 100000 nM T83193 C10QZR 118720710 EC50 = 8000 nM T83193 C4C6IY 118720711 EC50 = 1100 nM T83193 CC3JI2 118720712 EC50 = 16200 nM T83193 CU41SM 118720713 EC50 = 2500 nM T83193 CMHI10 118720714 EC50 = 10700 nM T83193 CP51VQ 118720715 EC50 = 8700 nM T83193 CC2A4O 118720716 IC50 > 100000 nM T83193 CV58RZ 118720717 IC50 > 100000 nM T83193 CAS16Q 118720718 IC50 > 100000 nM T83193 C19AGC 118720719 IC50 > 100000 nM T83193 CDL9U8 118720720 IC50 > 100000 nM T83193 CE7Q3M 118720721 IC50 > 100000 nM T83193 CG8JZ5 118720722 IC50 > 100000 nM T83193 C8XEA1 118720723 IC50 > 100000 nM T83193 CK9SH2 118720724 IC50 > 100000 nM T83193 CFBS82 118720725 EC50 = 430 nM T83193 CB17KL 118720726 IC50 > 100000 nM T83193 C9SD8T 118720727 EC50 = 1700 nM T83193 CI53FJ 118720728 EC50 = 8900 nM T83193 CH9WE1 118720729 EC50 = 6500 nM T83193 C8D9NZ 118720730 EC50 = 7800 nM T83193 C9S7AD 118720731 IC50 > 100000 nM T83193 CUR3X5 118720732 IC50 > 100000 nM T83193 CL0J1A 118720733 IC50 > 100000 nM T83193 CQF2M9 118723540 IC50 = 203000 nM T83193 C8P6NQ 118723541 IC50 = 10000 nM T83193 CCA4I7 118723542 IC50 = 19000 nM T83193 C5B8RU 118723543 IC50 = 48000 nM T83193 C8XMY5 118723544 IC50 = 70000 nM T83193 C8NB1I 118723545 IC50 = 45000 nM T83193 CFH7X4 118723546 IC50 = 8000 nM T83193 CZDF29 118723547 IC50 = 13000 nM T83193 C1PM6B 118723548 IC50 = 6000 nM T83193 CPJL95 118723549 IC50 = 9000 nM T83193 CP3R7M 118730332 Ki = 0.9 nM T83193 C5WG9H 118730333 Ki = 1.1 nM T83193 CN63MX 118730445 Ki = 3 nM T83193 CZTH58 118735927 IC50 > 10000 nM T83193 CEXG34 118735928 IC50 = 4300 nM T83193 CS7P9K 118735929 IC50 > 10000 nM T83193 C38JDV 118737608 Ki = 40.3 nM T83193 C6C9EF 121304827 IC50 > 3000 nM T83193 CAYH20 121364823 EC50 = 5.05 nM T83193 C1XNR3 121513880 IC50 > 10000 nM T83193 CB08PN 122193011 Ki = 3.9 nM T83193 C9NE4L 122193012 Ki = 2 nM T83193 C2S4NZ 122193013 Ki = 0.7 nM T83193 CIG7L0 122193014 Ki = 0.8 nM T83193 CBL0C9 122193015 Ki = 0.5 nM T83193 CZY7I1 122193016 Ki = 0.5 nM T83193 C6RL2A 122193017 Ki = 1.9 nM T83193 COU4P1 122193018 Ki = 2.3 nM T83193 CWS0T6 122193019 Ki = 1.8 nM T83193 C9UC0H 122193020 Ki = 1.4 nM T83193 CL93XU 122193022 Ki = 0.03 nM T83193 C7NEC1 122193023 Ki = 0.5 nM T83193 C2QW9Y 122193024 Ki = 13.9 nM T83193 C67NQR 122193025 Ki = 0.5 nM T83193 CM1V9A 122193026 Ki = 1.1 nM T83193 C9Y3XG 122194129 Ki = 0.9 nM T83193 C85KXR 122194130 Ki = 2.3 nM T83193 C9Q6PD 122194131 Ki = 3.2 nM T83193 CPS08K 122194132 Ki = 0.4 nM T83193 C2FYP9 122194133 Ki = 0.6 nM T83193 CE0H9Q 122194238 Ki = 1.2 nM T83193 CKW14B 122194340 Ki = 0.4 nM T83193 C2XOI4 122194341 Ki = 0.4 nM T83193 CA5HR7 122489394 IC50 > 20000 nM T83193 C74SXU 127025660 EC50 = 3970 nM T83193 C01GNA 127026006 Ki = 2.32 nM T83193 C2N8AP 127026007 Ki = 6 nM T83193 CWFH46 127026247 Ki = 0.76 nM T83193 CZV1H2 127026248 Ki = 0.71 nM T83193 CZ76GR 127026249 Ki = 0.9 nM T83193 C0CT8B 127026250 Ki = 1.65 nM T83193 CZGX18 127026253 Ki = 3.28 nM T83193 C4P3JA 127026320 Ki = 7.3 nM T83193 C6TJE7 127026548 IC50 > 10000 nM T83193 CY5L2R 127026553 EC50 = 320 nM T83193 C96DOK 127026858 IC50 > 10000 nM T83193 C63FIE 127026927 Ki = 1.29 nM T83193 CL2J1U 127026928 Ki = 2.14 nM T83193 C04QRN 127026929 Ki = 1.85 nM T83193 CE8BQ3 127026930 Ki = 1.56 nM T83193 C7QPD9 127027216 IC50 > 10000 nM T83193 C5EZR8 127027217 EC50 = 1530 nM T83193 CYWS67 127027218 EC50 = 1000 nM T83193 C7ST5H 127027220 EC50 = 1460 nM T83193 C32MSO 127027221 IC50 = 34 nM T83193 CP6UK0 127027222 IC50 > 10000 nM T83193 C4RGC5 127027223 IC50 > 10000 nM T83193 C2ESL3 127027524 EC50 = 310 nM T83193 CX8K3W 127027525 EC50 = 1990 nM T83193 C5IJF2 127027526 EC50 = 2250 nM T83193 C29BWY 127027527 EC50 = 370 nM T83193 CVHZ19 127028102 IC50 = 1950 nM T83193 CG5S3H 127028103 IC50 = 41 nM T83193 CBH98Z 127028104 EC50 = 660 nM T83193 CBI86M 127028105 EC50 = 170 nM T83193 CT4EN3 127028474 EC50 = 520 nM T83193 CO6C7E 127028475 IC50 > 10000 nM T83193 CXS10T 127028476 IC50 > 10000 nM T83193 CS1RH4 127028477 IC50 > 10000 nM T83193 C2J4XO 127028758 EC50 = 22 nM T83193 CE2NK5 127028759 EC50 = 20 nM T83193 C4RSM7 127028760 EC50 = 4230 nM T83193 C13LHT 127028800 IC50 > 10000 nM T83193 C7U3MP 127029033 IC50 = 1390 nM T83193 CD2TB1 127029037 IC50 > 10000 nM T83193 CHRE59 127029038 IC50 = 4130 nM T83193 C5BX0A 127029039 IC50 = 8110 nM T83193 CAP7Y6 127029097 Ki = 2.3 nM T83193 C4E8QM 127029371 Ki = 0.54 nM T83193 CS3ER8 127029372 Ki = 100 nM T83193 CB8S2H 127029373 Ki = 27.6 nM T83193 CXI5F8 127029645 Ki = 25 nM T83193 CO2NT6 127029646 Ki = 11.9 nM T83193 C4MYB0 127029647 Ki = 6.19 nM T83193 CI80PT 127029648 Ki = 3.13 nM T83193 C62AWV 127034988 IC50 = 173 nM T83193 CZU6J0 127034993 IC50 = 28 nM T83193 CCJ8G9 127035008 IC50 = 370 nM T83193 C4ORS9 127035153 IC50 = 783 nM T83193 C82YBF 127035453 IC50 = 653 nM T83193 C5MN6C 127035454 IC50 = 549 nM T83193 CB4E5T 127035456 IC50 = 67 nM T83193 CW6H7Q 127035457 IC50 = 75 nM T83193 CPFS58 127035458 IC50 = 125 nM T83193 C07TUH 127035459 IC50 = 136 nM T83193 C9V3CE 127035617 IC50 = 347 nM T83193 CFZ95J 127035618 IC50 = 325 nM T83193 CQ4MH9 127035822 IC50 = 127 nM T83193 C30NVR 127035823 IC50 = 239 nM T83193 CH94SE 127035824 IC50 = 381 nM T83193 CAMI26 127035825 IC50 = 24 nM T83193 C8Q1SD 127036261 IC50 = 591 nM T83193 CHB49J 127036589 IC50 = 359 nM T83193 CR16XZ 127036590 IC50 = 86 nM T83193 CDP78L 127037569 IC50 = 403 nM T83193 C6CXG5 127037570 IC50 = 38 nM T83193 C5YZ1L 127049919 Ki = 18.7 nM T83193 C3ZWT2 127049920 Ki = 28.1 nM T83193 CBU1F8 127049921 Ki = 59 nM T83193 C0ZC8V 127049922 Ki = 490 nM T83193 C2RHZ8 127050730 Ki = 83 nM T83193 C74JPG 127050731 Ki = 210 nM T83193 CJZ7Y8 132569635 IC50 > 10000 nM T83193 CMD64J 132942889 IC50 = 49700 nM T83193 C7Y4FE 132942890 IC50 = 68500 nM T83193 CD8P7C 132942891 IC50 = 53000 nM T83193 C4XK9Z 132942893 IC50 = 68900 nM T83193 CTJF87 134134782 IC50 > 10000 nM T83193 C3TW0A 134374895 IC50 > 30000 nM T83193 CPA8R4 135373178 EC50 = 200 nM T83193 CMX3A6 135373212 EC50 = 320 nM T83193 CB3FD2 135373234 EC50 = 370 nM T83193 CXZ6F7 135373249 IC50 = 930 nM T83193 CC5DJ8 135373260 IC50 = 90 nM T83193 CYHW05 135373273 EC50 = 450 nM T83193 CE0DR3 135373275 EC50 = 40 nM T83193 C28RFL 135373302 EC50 = 410 nM T83193 CU8PR6 135373307 EC50 = 330 nM T83193 C4PH1D 135373311 EC50 = 40 nM T83193 CR7S8O 135373364 EC50 = 90 nM T83193 CL87FA 135373389 EC50 = 170 nM T83193 CLAY04 135373392 EC50 = 140 nM T83193 C4N7MS 135373395 IC50 = 1340 nM T83193 C0R8IK 135433889 IC50 = 13 nM T83193 C0Y7WF 135444669 IC50 = 50 nM T83193 C3O9XM 135465551 IC50 = 14 nM T83193 C67MSV 135474346 IC50 = 31 nM T83193 C4EN0K 135492547 IC50 = 12 nM T83193 C1IV8U 136027059 IC50 = 1343 nM T83193 C7BW3K 136094797 IC50 = 487 nM T83193 C0GIS5 136094798 IC50 = 557 nM T83193 C73EKQ 136094799 IC50 = 40 nM T83193 C63WKI 136094800 IC50 = 133 nM T83193 C4LS1T 136094801 IC50 = 42 nM T83193 CF18ME 136094802 IC50 = 144 nM T83193 CPQ7Y1 136094803 IC50 = 23 nM T83193 CQ9EP5 136094804 IC50 > 1000 nM T83193 CF3KG8 136094805 IC50 = 82 nM T83193 CIS4K7 136094806 IC50 = 201 nM T83193 CA8MI2 136094807 IC50 = 216 nM T83193 C41JRM 136094808 IC50 = 286 nM T83193 C4Z3GW 136094809 IC50 > 1000 nM T83193 CV40RL 136094810 IC50 = 100 nM T83193 CPNF93 136094811 IC50 = 37 nM T83193 CZY5X9 137007154 EC50 = 6900 nM T83193 CHO40Y 137007155 EC50 = 5500 nM T83193 C0NU7J 137007156 EC50 = 37500 nM T83193 CF5IN0 137007157 IC50 > 100000 nM T83193 CX52EQ 137634042 Ki = 6.7 nM T83193 CW35LN 137634053 Ki = 112 nM T83193 CGME50 137634139 Ki = 51.8 nM T83193 C35VLF 137634200 Ki = 1.9 nM T83193 CG6E3D 137634936 Ki = 1.5 nM T83193 C3NYE0 137636166 Ki = 4.1 nM T83193 CJH2V9 137637559 IC50 > 30000 nM T83193 CJS75L 137639554 Ki = 3.4 nM T83193 CZ4SA7 137640006 Ki = 0.7 nM T83193 CFMN82 137642621 Ki = 8.5 nM T83193 CE17JM 137643454 Ki = 17.1 nM T83193 CGT02Z 137644147 Ki = 2.8 nM T83193 CZM60X 137644630 Ki = 6 nM T83193 CXC8H3 137646362 Ki = 4.4 nM T83193 CL97NH 137646641 Ki = 4 nM T83193 C46HTO 137647720 Ki = 5.9 nM T83193 CNB4W7 137648188 Ki = 1 nM T83193 C7T5UR 137649873 Ki = 6 nM T83193 CHB60E 137649975 Ki = 89.2 nM T83193 CR35QL 137649976 Ki = 3.2 nM T83193 CZ4B1S 137650495 Ki = 3.4 nM T83193 C0K7PN 137650773 Ki = 0.3 nM T83193 C6R5OF 137651359 Ki = 9.8 nM T83193 CJ9L0P 137652512 Ki = 3.5 nM T83193 C15RPF 137652934 Ki = 2.5 nM T83193 C9UWO7 137654328 Ki = 3.1 nM T83193 CQ5K4S 137654340 Ki = 0.63 nM T83193 C21JIB 137654381 Ki = 3.8 nM T83193 CC5HF6 137654715 Ki = 0.6 nM T83193 C6GWK3 137656096 Ki = 6.2 nM T83193 CFA87N 137656645 Ki = 7.4 nM T83193 CQO4K3 137656714 Ki = 3.1 nM T83193 CX5BP4 137656937 Ki = 0.8 nM T83193 C6WM9Z 137657008 Ki = 0.3 nM T83193 CK7SZ1 137657211 Ki = 0.1 nM T83193 CRL18A 137658691 Ki = 8.1 nM T83193 C0QTE6 137659796 Ki = 3.8 nM T83193 CW1IL7 137660362 Ki = 0.5 nM T83193 C32YDL 137660439 Ki = 2.9 nM T83193 C2KX3V 137661020 IC50 > 30000 nM T83193 CY46UQ 137661067 Ki = 0.8 nM T83193 C39HPA 137661261 IC50 > 10000 nM T83193 C8FWK9 137662018 Ki = 1.2 nM T83193 CRI14T 137662297 Ki = 36.4 nM T83193 CEK6B1 139300630 IC50 > 10000 nM T83193 CD4OJ3 141507741 IC50 = 12.8 nM T83193 CC7PG9 141507742 IC50 = 76 nM T83193 C2OGN0 141507743 IC50 = 46.8 nM T83193 CGN93F 141507744 IC50 = 12.2 nM T83193 CPBZ17 141507745 IC50 = 39.6 nM T83193 C8ZM7G 141507746 IC50 = 14 nM T83193 C70TDA 141507748 IC50 = 250.3 nM T83193 C6X2BP 141507750 IC50 = 125.2 nM T83193 CZI7O3 141507751 IC50 = 12.3 nM T83193 CG08HC 141507753 IC50 = 16.4 nM T83193 C7M1DR 141507754 IC50 = 80.3 nM T83193 C0FE1B 141507755 IC50 = 45.2 nM T83193 C3OA9W 141507756 IC50 = 10.2 nM T83193 CP3BC5 141507757 IC50 = 36.4 nM T83193 C98MWI 141507758 IC50 = 37 nM T83193 CW9A4T 141507759 IC50 = 22 nM T83193 CU1HB0 141507760 IC50 = 40.7 nM T83193 C3RX5K 141507761 IC50 = 43.5 nM T83193 CQ0K8F 141507762 IC50 = 37.6 nM T83193 C6NA4O 141507763 IC50 = 12.7 nM T83193 CK53FW 141507764 IC50 = 46 nM T83193 CD69ZJ 141507765 IC50 = 136.2 nM T83193 C2C1ND 141507767 IC50 = 47.1 nM T83193 CF6XQ0 141507768 IC50 = 70.3 nM T83193 C9D1QP 141507769 IC50 = 40.5 nM T83193 CJ7I0E 141507770 IC50 = 14 nM T83193 CIC73G 141756420 IC50 = 243 nM T83193 C3VHP9 141756421 IC50 = 385 nM T83193 C19VLF 141756424 IC50 = 495 nM T83193 CD7OE4 141756426 IC50 = 2156 nM T83193 CG4P5R 141756427 IC50 = 1122 nM T83193 CM4IX7 141756430 IC50 = 3489 nM T83193 C81AOD 141756431 IC50 = 1674 nM T83193 C24LJR 141756433 IC50 = 121 nM T83193 C2PZB6 145952645 Ki = 2.3 nM T83193 CJ1WT7 145952872 IC50 = 200 nM T83193 C43IUN 145953312 IC50 = 98 nM T83193 CU71FI 145953315 IC50 = 1800 nM T83193 CO9JR6 145953318 IC50 = 72 nM T83193 CWFX19 145954238 IC50 = 95 nM T83193 C4ZH3R 145954944 IC50 = 510 nM T83193 CQ0T2U 145954951 IC50 = 150 nM T83193 CZX10U 145955162 IC50 = 29 nM T83193 CEFH61 145955415 IC50 = 1300 nM T83193 CX0IJ3 145955646 IC50 = 890 nM T83193 CUT2Z8 145955878 Ki = 3.2 nM T83193 C15VSY 145960411 Ki = 0.7 nM T83193 C5RLE1 145960771 IC50 = 470 nM T83193 C52ALB 145960801 Ki = 0.2 nM T83193 CU8L7X 145960890 IC50 = 150 nM T83193 CG3U1B 145961025 IC50 = 820 nM T83193 CB7L9N 145961796 Ki = 0.3 nM T83193 CDYL02 145961805 Ki = 2.4 nM T83193 C1INS9 145962051 IC50 = 700 nM T83193 CJ9BA4 145962156 IC50 = 580 nM T83193 CSCL29 145962213 IC50 = 140 nM T83193 C0O2DH 145962509 Ki = 1.6 nM T83193 CIHR57 145962782 IC50 = 23 nM T83193 CVH7K8 145962832 IC50 = 150 nM T83193 C5TE0L 145962994 IC50 = 320 nM T83193 CG2DY1 145963166 IC50 = 73 nM T83193 CXCD86 145963177 IC50 = 530 nM T83193 CCUD75 145963228 IC50 = 86 nM T83193 CI34EM 145963457 IC50 = 480 nM T83193 C2T1CI 145965659 Ki = 819 nM T83193 CTMX69 145968194 EC50 = 3690 nM T83193 C1N5FP 145968965 IC50 = 81.9 nM T83193 C8C5OW 145969594 IC50 = 10.6 nM T83193 CQL1I9 145972802 Ki = 0.1 nM T83193 C9ME8W 145974998 Ki = 8 nM T83193 C80UTE 145976266 Ki = 50.2 nM T83193 C0WR3F 145976623 Ki = 5.1 nM T83193 C1ZA4F 145977088 IC50 = 25.7 nM T83193 C6KW1F 145983017 IC50 = 297 nM T83193 C4DPI9 145983348 Ki = 20 nM T83193 C5OL8C 145983461 Ki = 66.5 nM T83193 C40INH 145983507 IC50 > 50000 nM T83193 CS9Z6B 145983717 IC50 = 46 nM T83193 CH9AW8 145983743 IC50 = 25 nM T83193 CYVP70 145983755 IC50 = 352 nM T83193 C2TQK7 145983963 Ki = 7.4 nM T83193 CYGR61 145983976 Ki = 5.3 nM T83193 C79POF 145984006 Ki = 0.1 nM T83193 CJ9X5Q 145984060 IC50 = 684 nM T83193 C6H0QM 145984205 IC50 > 100000 nM T83193 C2AO8L 145984443 IC50 = 20 nM T83193 CO54SW 145984817 Ki = 51.9 nM T83193 CB61OL 145985025 IC50 = 458 nM T83193 CL8WN5 145985126 Ki = 21 nM T83193 C0YQ6D 145985141 Ki = 2.4 nM T83193 CWZ1U5 145985255 Ki = 26.4 nM T83193 CF6DU3 145985290 IC50 = 621 nM T83193 C5WVH1 145985756 IC50 > 100000 nM T83193 CC4Q1B 145985949 EC50 = 4900 nM T83193 C2MAB1 145986122 EC50 = 1800 nM T83193 C6EF2M 145986126 IC50 = 461 nM T83193 C4EFS1 145986233 IC50 = 33 nM T83193 CXJH67 155510378 Ki = 0.67 nM T83193 C93ETV 155511833 IC50 = 89 nM T83193 CXS52I 155512061 IC50 = 204 nM T83193 C3E0TA 155512687 IC50 = 22573 nM T83193 CG6MB4 155513334 IC50 = 232 nM T83193 CX4Z3F 155513383 Ki = 0.95 nM T83193 CI65OP 155513602 Ki = 10.8 nM T83193 CYRX70 155515945 Ki = 12.3 nM T83193 C05DLO 155517206 IC50 = 75 nM T83193 CBHC08 155517653 IC50 = 341 nM T83193 CZS69J 155518412 IC50 = 27071 nM T83193 CZ79SG 155518694 IC50 = 1543 nM T83193 CT93LK 155520217 EC50 = 43.7 nM T83193 CVL45A 155523755 IC50 = 788 nM T83193 CY8XL4 155524179 Ki = 7.33 nM T83193 CS0LP7 155525545 Ki = 62 nM T83193 CSL9T1 155525842 EC50 = 31.3 nM T83193 C3IG2A 155526856 IC50 = 1195 nM T83193 CEJI39 155527289 Ki = 14.1 nM T83193 CA16DV 155528800 IC50 = 112 nM T83193 C3NEY4 155530370 IC50 = 394 nM T83193 C0W2GI 155531907 IC50 = 12572 nM T83193 C7QW0U 155532849 IC50 = 1878 nM T83193 C38MQU 155533274 IC50 = 19416 nM T83193 CG6C1I 155535201 Ki = 0.46 nM T83193 CG27DS 155537117 IC50 = 494 nM T83193 CD34OK 155537741 IC50 = 108 nM T83193 CUX51M 155538186 EC50 = 85.9 nM T83193 C8EQ5U 155538902 IC50 = 81600 nM T83193 C6IJA4 155539728 Ki = 1159 nM T83193 CS79MX 155547713 IC50 = 2531 nM T83193 CL36YR 155548389 Ki = 15.3 nM T83193 CPT0Q4 155553946 IC50 = 4945 nM T83193 CN61OU 155554804 IC50 = 1217 nM T83193 CEY91R 155556936 IC50 = 416 nM T83193 CB3DO5 155556993 Ki = 27.9 nM T83193 CHU9L6 155559739 Ki = 1.67 nM T83193 C8I3RS 155562884 Ki = 16.4 nM T83193 D00AII 5281727 IC50 > 10000 nM T83193 D00AJB 73255 IC50 = 50000 nM T83193 D00HCI 1598 EC50 = 129000 nM T83193 D00RDS 797382 Ki = 24 nM T83193 D00XZZ 4286311 EC50 = 300 nM T83193 D00ZWU 1860395 Ki = 53 nM T83193 D01DIT 5283446 EC50 = 630 nM T83193 D01WDS 44450288 Ki = 156 nM T83193 D02GOH 6604822 EC50 = 26 nM T83193 D03HFM 42617984 EC50 = 23 nM T83193 D03LVL 53464483 IC50 > 25000 nM T83193 D03SCD 44448616 EC50 > 100000 nM T83193 D03SJY 24749270 IC50 = 760 nM T83193 D04AMC 11559610 EC50 = 260 nM T83193 D04ECZ 42617986 EC50 = 13 nM T83193 D04XXE 73489 IC50 = 170000 nM T83193 D05APW 46890602 IC50 = 7 nM T83193 D05NTO 5149140 IC50 = 10 nM T83193 D06CDW 3035862 Ki = 0.12 nM T83193 D06MRN 44450313 Ki = 15 nM T83193 D07BKU 11451659 IC50 = 14 nM T83193 D07LCG 44450366 Ki = 6272 nM T83193 D07MBC 5283454 EC50 = 40 nM T83193 D07YQG 5282105 EC50 = 50 nM T83193 D08KRX 4375060 Ki = 980 nM T83193 D08KYH 44450322 Ki = 70 nM T83193 D08WAW 2796370 Ki = 421 nM T83193 D09AZO 44416783 IC50 = 2585 nM T83193 D09BEW 44450379 Ki = 15000 nM T83193 D09OSN 151253 IC50 > 10000 nM T83193 D09SXM 24768211 IC50 = 73 nM T83193 D09WYF 44450365 EC50 > 5000 nM T83193 D0A9PS 5281969 EC50 = 15.8 nM T83193 D0BB7F 44450355 Ki = 72 nM T83193 D0C3XF 44450381 Ki = 607 nM T83193 D0D0DW 11302766 IC50 = 170 nM T83193 D0D4SO 3904199 Ki = 2080 nM T83193 D0D6MC 1150897 IC50 > 20000 nM T83193 D0D6OH 104895 EC50 = 10 nM T83193 D0D7QH 6449767 EC50 = 0.5012 nM T83193 D0D9MW 4298023 Ki = 60 nM T83193 D0DJ6G 44450356 Ki = 29 nM T83193 D0DL4Y 22020504 IC50 = 51 nM T83193 D0DY4E 11339118 IC50 = 65 nM T83193 D0E2XP 24749267 IC50 = 1820 nM T83193 D0E4FJ 5283381 IC50 = 35 nM T83193 D0F1UD 4589192 IC50 = 9100 nM T83193 D0F4NA 1019468 IC50 = 330 nM T83193 D0FF6S 16038374 IC50 > 10000 nM T83193 D0G2EQ 42617990 EC50 = 47 nM T83193 D0G8BN 2733484 IC50 = 4 nM T83193 D0H6GW 44450346 Ki = 1740 nM T83193 D0H6TX 24768210 IC50 = 749 nM T83193 D0J3VX 10248092 IC50 = 91 nM T83193 D0J7CR 42617983 EC50 = 610 nM T83193 D0K7QP 44591633 EC50 = 19 nM T83193 D0K8MN 44448617 EC50 = 10000 nM T83193 D0L9DR 9951636 IC50 = 49 nM T83193 D0M7NA 25224408 IC50 = 21 nM T83193 D0N2QH 6324614 Ki = 5.87 nM T83193 D0N8EI 44450336 IC50 = 66 nM T83193 D0O9NE 5388063 IC50 > 10000 nM T83193 D0P7VQ 9929425 IC50 = 0.18 nM T83193 D0Q0XV 44591632 EC50 = 180 nM T83193 D0Q2ZO 44450380 Ki = 546 nM T83193 D0Q4GB 637566 IC50 > 100000 nM T83193 D0Q8QH 11638703 EC50 = 400 nM T83193 D0R7QF 42617989 EC50 = 2400 nM T83193 D0R8XX 24749271 IC50 = 740 nM T83193 D0SH1L 10473280 IC50 = 600 nM T83193 D0T3CP 11645841 EC50 = 320 nM T83193 D0T8DR 44450347 IC50 = 150 nM T83193 D0U5LL 2543 EC50 = 6200 nM T83193 D0W3VM 11472986 IC50 = 11 nM T83193 D0W6TX 7927254 IC50 = 280 nM T83193 D0W7XR 11507802 IC50 > 100000 nM T83193 D0WK3N 44450300 Ki = 23 nM T83193 D0X7AM 10295883 EC50 = 8 nM T83193 D0X8XU 24768203 IC50 = 2580 nM T83193 D0XO2G 680502 IC50 = 150 nM T83193 D0Y1MM 11710300 EC50 = 250 nM T83193 D0Y7QY 5885566 IC50 = 330 nM T83193 D0Y9EU 3884807 Ki = 3520 nM T83193 D0Z1NH 42617985 EC50 = 150 nM T35465 D01KKQ 135400182 IC50 = 6.3 nM T35465 D02LWU 148121 IC50 = 0.69 nM T35465 D0SV8E 126941 IC50 = 12 nM T35465 D0Y4GO 135410875 IC50 = 138 nM T35465 CO2DY5 11247965 Ki = 280 nM T35465 C8Q6ZT 11248313 Ki = 1100 nM T35465 CM4Z7A 44421498 Ki = 530 nM T35465 CPM3L5 67092576 IC50 = 54 nM T35465 CTK64O 67092918 IC50 > 1000 nM T35465 C87FBU 135455948 IC50 = 59.8 nM T35465 CF8D5O 135465664 IC50 > 1000 nM T35465 C9Z4ES 135567027 IC50 > 1000 nM T35465 C14LTO 135567028 IC50 > 1000 nM T35465 CF39AI 135567029 IC50 = 101 nM T35465 C8N7ES 135567030 IC50 > 1000 nM T35465 CFE2O7 135567034 IC50 = 197 nM T35465 C8KVP5 135567035 IC50 = 189 nM T35465 CSQX75 135567163 IC50 = 510 nM T35465 CQF8P5 135800109 IC50 = 304 nM T35465 CL8VN5 136015502 IC50 = 116 nM T35465 CR7UY3 136044173 IC50 > 1000 nM T35465 C0Q5FI 136044174 IC50 > 1000 nM T35465 CGX68Y 136044175 IC50 > 1000 nM T35465 C4C9FN 136044176 IC50 > 1000 nM T35465 CIPD35 136044177 IC50 > 1000 nM T35465 CZG8W6 136059167 IC50 = 634 nM T35465 CZC95Y 136059168 IC50 > 1000 nM T35465 CG2ID9 136059169 IC50 > 1000 nM T35465 C2WH0S 136059178 IC50 > 1000 nM T35465 CB3GL7 136059191 IC50 > 1000 nM T35465 CCHG08 136059192 IC50 > 1000 nM T35465 C4Q1HF 136180345 IC50 = 38.3 nM T35465 CDC83K 136180346 IC50 = 243.2 nM T35465 CF7NW6 136180347 IC50 > 1000 nM T35465 CPH52E 137150145 IC50 > 1000 nM T35465 C9XD1M 137150146 IC50 > 1000 nM T35465 CHDB56 137150160 IC50 > 1000 nM T35465 CMKA64 155517044 IC50 = 808 nM T35465 CCL3Y9 155518053 IC50 = 66.2 nM T35465 C91SVN 155519837 IC50 = 641 nM T35465 CO7BN6 155524531 IC50 > 1000 nM T35465 CT70WU 155530762 IC50 = 213 nM T35465 CX42MF 155532591 IC50 > 1000 nM T35465 CFU98A 155534971 IC50 = 642 nM T35465 C4K2RU 155538415 IC50 > 1000 nM T35465 C27BIX 155539477 IC50 > 1000 nM T35465 C6S7OC 155548982 IC50 = 62 nM T35465 CX3K8F 155549935 IC50 > 1000 nM T35465 CJ0MK5 155554671 IC50 = 468 nM T35465 CYQ0I9 155555353 IC50 = 783 nM T46828 D01AZG 5073 Ki = 1000 nM T46828 D01FFA 72301 Ki = 305 nM T46828 D01ZII 2726 Ki = 172 nM T46828 D03KQF 4011 Ki = 429 nM T46828 D05XGO 11154555 Ki = 7900 nM T46828 D0B0CP 667467 Ki = 9 nM T46828 D0CQ0Z 33630 Ki = 125 nM T46828 D0D1AL 3559 Ki = 38 nM T46828 D0G8NN 119570 Ki > 10000 nM T46828 D0H3HM 60795 Ki > 1000 nM T46828 D0H7KF 5002 Ki > 1000 nM T46828 D0KS6W 7077 Ki = 414 nM T46828 D0P5SA 3372 Ki = 21 nM T46828 D0R9EQ 5095 Ki = 41211 nM T46828 D0T7OW 681 EC50 = 2 nM T46828 D0V4QS 135398745 Ki = 90 nM T46828 D0Y5UG 2160 Ki = 170 nM T46828 D0Z1RV 135398737 Ki = 198 nM T46828 D0N1HW 5311200 Ki > 10000 nM T46828 D0Y6HW 107930 Ki = 2 nM T46828 D07YLK 4350931 Ki = 7.5 nM T46828 D02DHU 1218 EC50 = 1.4 nM T46828 D06DZI 107780 Ki > 10000 nM T46828 D0M7LV 5761 Ki = 340 nM T46828 D0OU7P 1242 Ki = 124 nM T46828 D0OW1R 9802631 Ki > 10000 nM T46828 C5H9CN 9287 Ki > 10000 nM T46828 C9E6DA 21171 Ki = 62.1 nM T46828 C17TDE 23269 Ki > 10000 nM T46828 CBJ5R0 65340 Ki = 1023.29 nM T46828 C6CU1T 70515 Ki > 10000 nM T46828 CPZ5N6 98358 Ki > 10000 nM T46828 C1ND9W 161665 Ki = 242 nM T46828 C09JTU 199798 Ki > 10000 nM T46828 C5RC4G 231915 Ki > 10000 nM T46828 CYO3R2 300430 Ki > 10000 nM T46828 CG2JX9 440229 Ki = 9.5 nM T46828 CQZ4A9 636934 Ki > 10000 nM T46828 CD7P8Y 763194 Ki > 10000 nM T46828 C6QLR0 763343 Ki > 10000 nM T46828 CLR75J 763625 Ki = 2059 nM T46828 C5SXQ1 763774 Ki = 3523 nM T46828 C9IK2J 792265 Ki > 10000 nM T46828 C13TYL 792460 Ki > 10000 nM T46828 C4AY9X 792584 Ki > 10000 nM T46828 CVTP62 1811569 Ki > 10000 nM T46828 C4TB0I 3036864 Ki = 0.48 nM T46828 C64CZV 3038494 Ki = 1223 nM T46828 C82GMT 3246443 Ki = 15.1 nM T46828 C0U6EW 3504099 Ki > 10000 nM T46828 C6AQP8 5249952 Ki = 112 nM T46828 C9AZ2I 5249956 Ki = 3.09 nM T46828 CO3N1A 6440792 IC50 = 0.15 nM T46828 C8QM7B 6852376 Ki = 245.47 nM T46828 C7EZ2L 9859861 Ki > 10000 nM T46828 C5WYN4 9865858 Ki > 1000 nM T46828 C3DB5H 9884781 Ki > 3000 nM T46828 C6WY0D 9891901 Ki > 10000 nM T46828 CYWQ50 9906447 Ki > 10000 nM T46828 CP41ZO 9992499 Ki = 337 nM T46828 CZKG96 10200496 Ki = 16.6 nM T46828 C6J2ZL 10402378 Ki = 1.8 nM T46828 C2B0IU 10421236 Ki > 10000 nM T46828 COV85C 10472143 Ki = 400 nM T46828 CPI5M7 10476504 Ki = 3700 nM T46828 CEF2O6 10478367 Ki > 10000 nM T46828 CRI50E 10885636 IC50 = 988 nM T46828 CNP08C 10891703 Ki > 10000 nM T46828 CX65PW 10907460 IC50 = 1450 nM T46828 CQ62UO 10918307 IC50 = 3660 nM T46828 CNB39C 10947658 Ki = 1000 nM T46828 CJC9K4 11005810 IC50 = 513 nM T46828 CFJG64 11059058 IC50 = 4890 nM T46828 CG41BK 11071079 IC50 = 1550 nM T46828 C7DE0U 11113605 IC50 = 3020 nM T46828 CVE8T3 11121216 Ki = 590 nM T46828 CUD5A0 11134444 Ki = 1756 nM T46828 C3NEM0 11151473 Ki = 9600 nM T46828 C5JS0L 11151831 Ki = 12000 nM T46828 C4FTD9 11153135 Ki = 83000 nM T46828 C3Q9UG 11154178 Ki = 13 nM T46828 CN06GJ 11186895 Ki = 313 nM T46828 C8FKS6 11198948 Ki = 5900 nM T46828 C7MY8T 11210215 Ki = 19000 nM T46828 CVT04Q 11221294 Ki = 9000 nM T46828 C8RJ3D 11223303 Ki = 7.1 nM T46828 CKX06B 11235174 Ki = 5.8 nM T46828 C1Z4WT 11246806 Ki = 26000 nM T46828 CM72YX 11269330 Ki = 10.5 nM T46828 CUJ2R7 11280344 Ki > 10000 nM T46828 CF1C7M 11290269 Ki = 8300 nM T46828 CLZ9S1 11290688 Ki = 7200 nM T46828 CG95WP 11301268 Ki = 71000 nM T46828 C45WLN 11324023 Ki = 16000 nM T46828 CXWH42 11358377 Ki = 1812 nM T46828 CY24NV 11374299 Ki = 5.9 nM T46828 CP3Y2E 11394805 Ki = 32000 nM T46828 C6O9QT 11405458 Ki = 7700 nM T46828 CT32OJ 11406143 Ki = 620 nM T46828 C95WMQ 11415988 Ki = 7600 nM T46828 C1OUA4 11416809 Ki = 20000 nM T46828 CKQ6F7 11416811 Ki = 16000 nM T46828 CF2V6Y 11438636 Ki = 16000 nM T46828 CBN91Q 11439190 Ki = 89 nM T46828 C6A0EF 11439436 Ki = 15000 nM T46828 CD4UV2 11441173 Ki = 54000 nM T46828 C37RKD 11449266 Ki = 19000 nM T46828 CS34HD 11449669 Ki = 19000 nM T46828 C4YT6M 11450584 Ki = 9600 nM T46828 C86CJB 11451022 Ki > 10000 nM T46828 CB3P6S 11452916 Ki = 5.6 nM T46828 CK39HZ 11486421 Ki = 3.3 nM T46828 CTU1Z7 11488247 Ki = 1.2 nM T46828 CKV25P 11493746 Ki = 1.2 nM T46828 CR1HO4 11500181 Ki > 10000 nM T46828 CAU1R7 11500677 Ki = 1050 nM T46828 CQ5IN9 11522339 Ki = 10.4 nM T46828 CC6U7R 11522476 Ki = 2610 nM T46828 C75YUO 11536580 Ki > 10000 nM T46828 C2JT3I 11536995 Ki = 54.6 nM T46828 CN3W7S 11543350 Ki > 10000 nM T46828 C8X0EM 11543992 Ki > 10000 nM T46828 C0AN1Y 11551474 Ki > 10000 nM T46828 C7S2WZ 11558055 Ki = 1.5 nM T46828 CM8G3B 11558247 Ki = 39.5 nM T46828 C4HDA6 11558324 Ki > 10000 nM T46828 C8GK0U 11566745 Ki = 2.32 nM T46828 CP8MF4 11573628 Ki = 3.1 nM T46828 C1TBC8 11573806 Ki = 11.5 nM T46828 C5Q8XM 11595240 Ki = 0.98 nM T46828 CFC25K 11601627 Ki > 10000 nM T46828 C9D7OU 11616435 Ki > 10000 nM T46828 CN1P4I 11623343 Ki = 0.54 nM T46828 CIZ53S 11623652 Ki > 10000 nM T46828 CS4CR7 11631304 Ki = 893 nM T46828 CMX4K8 11633643 Ki > 10000 nM T46828 CG1C3D 11637457 Ki = 15 nM T46828 CLZQ65 11644613 Ki > 10000 nM T46828 CHIW07 11652965 Ki > 10000 nM T46828 CO69ZI 11666419 Ki > 10000 nM T46828 CE34SW 11668495 Ki > 10000 nM T46828 CI26JH 11674133 Ki > 10000 nM T46828 CSQ4B1 11681599 Ki = 0.053 nM T46828 C06BEA 11694873 Ki > 10000 nM T46828 CRO95K 11695189 Ki > 10000 nM T46828 CN1SJ8 11696598 Ki > 10000 nM T46828 CDLW51 11701907 Ki > 10000 nM T46828 C0G1WQ 11709500 Ki > 10000 nM T46828 CI3N1K 11716230 Ki > 10000 nM T46828 CZ6NB8 11716438 Ki = 37.5 nM T46828 CZ7SJ2 11716449 Ki = 14.7 nM T46828 C9FTL5 11718008 Ki = 59 nM T46828 C7PVL8 11730467 IC50 = 1860 nM T46828 CA4W1P 11739113 Ki = 13000 nM T46828 CV91RG 11778580 Ki = 0.57 nM T46828 CH5T6L 11818686 Ki = 16000 nM T46828 CXLW54 11948707 Ki > 10000 nM T46828 C8JQL7 11957735 IC50 > 10000 nM T46828 C7NV4W 12068769 Ki > 10000 nM T46828 C4NWX9 12301195 Ki > 10000 nM T46828 CCG14E 13091356 Ki > 10000 nM T46828 CC74ND 13373172 Ki = 41.1 nM T46828 CI5Y6N 13611248 Ki > 10000 nM T46828 C7VAI1 15011772 Ki > 10000 nM T46828 C0G2EO 16007117 Ki = 73 nM T46828 CWMC70 16090814 Ki = 0.61 nM T46828 CP09RQ 16090821 Ki = 71.6 nM T46828 CZ2IS9 16660294 Ki > 10000 nM T46828 CGX0D5 16665071 Ki = 0.23 nM T46828 C7KP5T 17755866 Ki = 17 nM T46828 CX7VE8 17755867 Ki = 9.8 nM T46828 CUW8S4 17755868 Ki = 95 nM T46828 C3KA6Z 17755875 Ki > 10000 nM T46828 C4N1LS 17755991 Ki = 314 nM T46828 C6BE2Y 17755992 Ki > 10000 nM T46828 C10UQJ 17755999 Ki = 55 nM T46828 C6WO9X 17756101 Ki = 4.6 nM T46828 CI9RW0 17756102 Ki = 53 nM T46828 CDPT42 17756110 Ki > 10000 nM T46828 C0XG9B 17756212 Ki = 75 nM T46828 C6JQ1K 17756213 Ki = 69 nM T46828 CG5NT4 20035572 Ki > 10000 nM T46828 C94BPG 21460314 Ki > 10000 nM T46828 C3T5HF 21509921 Ki = 575.44 nM T46828 CFN81Q 21527771 Ki = 103 nM T46828 CH59WN 21533446 Ki = 113 nM T46828 CL5A2V 21554999 Ki > 10000 nM T46828 C61LUT 21555004 Ki > 10000 nM T46828 CAH39X 21564536 Ki > 10000 nM T46828 CO4C6M 23653115 Ki > 10000 nM T46828 CBUJ02 23653176 Ki = 202 nM T46828 CDH38J 23992579 Ki > 10000 nM T46828 C3W6DQ 25096873 IC50 > 1000 nM T46828 CX04LB 25142456 Ki = 7 nM T46828 C78HME 25212275 Ki = 265 nM T46828 CE6Z9I 25212276 Ki = 265 nM T46828 C4MRQ0 27842480 IC50 > 50000 nM T46828 CK3QD2 42625354 Ki = 80 nM T46828 CLH7Y0 42626289 Ki = 75.4 nM T46828 C5VTZ6 42626293 Ki = 313 nM T46828 CVG6X1 44209472 Ki = 2392 nM T46828 CD5AB7 44209480 Ki = 1451 nM T46828 C98VPM 44275670 Ki = 5.62 nM T46828 C1B4QL 44403095 Ki > 10000 nM T46828 C1YL7Z 44403098 Ki > 10000 nM T46828 CFV98A 44403101 Ki > 10000 nM T46828 C6OY9S 44403102 Ki > 10000 nM T46828 CH4SX6 44403105 Ki > 10000 nM T46828 C12FIH 44403106 Ki > 10000 nM T46828 C4LKC1 44404394 Ki > 10000 nM T46828 C3EJ4G 44404396 Ki > 10000 nM T46828 CO2H3T 44406799 Ki > 10000 nM T46828 CI70SN 44406862 Ki > 10000 nM T46828 C0R6PK 44406863 Ki > 10000 nM T46828 CDA3R0 44406866 Ki > 10000 nM T46828 CU52FA 44406881 Ki > 10000 nM T46828 CZ24HP 44408818 Ki = 7.2 nM T46828 C93NGH 44414299 Ki = 411 nM T46828 CU2FG6 44415569 Ki = 38 nM T46828 CDU6Y5 44415593 Ki = 105 nM T46828 CH0BY5 44415672 Ki = 7 nM T46828 CK59CO 44415689 Ki = 53 nM T46828 C7AZ5D 44415690 Ki = 31 nM T46828 CEVY54 44415704 Ki = 58 nM T46828 CY0QJ2 44427970 Ki = 510 nM T46828 C2AZ6B 44436300 Ki = 386 nM T46828 C30QMX 44436301 Ki = 230 nM T46828 C9AJ0D 44436302 Ki = 1132 nM T46828 C3NVL0 44436303 Ki > 10000 nM T46828 CREM27 44436304 Ki = 507 nM T46828 C53XYK 44436305 Ki = 1703 nM T46828 C2LF9K 44436306 Ki = 190 nM T46828 C9H8ST 44436307 Ki = 33.6 nM T46828 C7IBE2 44436308 Ki = 80.8 nM T46828 CBI86V 44439942 Ki = 3.6 nM T46828 C3HMI2 44439943 Ki = 0.39 nM T46828 C63PQV 44439944 Ki = 31.5 nM T46828 C2P4CI 44439945 Ki = 5.4 nM T46828 C12XGE 44456400 Ki > 10000 nM T46828 C16HEZ 44555445 Ki > 10000 nM T46828 CRCH48 44582675 Ki = 7419 nM T46828 CEJ4R8 44582676 Ki = 7398 nM T46828 CP6ZA9 44591012 Ki > 1000 nM T46828 CU37BO 44591098 Ki > 1000 nM T46828 CU48CL 44591099 Ki = 273 nM T46828 C7H9SE 44591134 Ki = 153 nM T46828 C6RLW0 44591135 Ki = 297 nM T46828 CYJ7P8 45379368 Ki > 10000 nM T46828 CU2CA7 45379369 Ki = 2.5 nM T46828 CT3K8Y 45379370 Ki = 10.3 nM T46828 CT3A1Q 45379373 Ki > 10000 nM T46828 C8TRE1 45379377 Ki = 1525 nM T46828 CML67J 45379515 Ki > 10000 nM T46828 CSV1P2 46216855 Ki = 1.9 nM T46828 CY7NM6 46227242 Ki > 10000 nM T46828 CR9S7B 46227243 Ki > 10000 nM T46828 C9A8FV 46227273 Ki > 10000 nM T46828 CL3KU2 46227284 Ki = 1508 nM T46828 CS4O6A 46227317 Ki = 185 nM T46828 CE1L6H 46227320 Ki > 10000 nM T46828 CSQ9D5 46227325 Ki = 1810 nM T46828 CDI10H 46231541 Ki = 3.9 nM T46828 C9KI4E 46231646 Ki = 8.3 nM T46828 C8SFI5 46231768 Ki = 7 nM T46828 C1EW4S 46231782 Ki = 3.7 nM T46828 C6JM5T 46231784 Ki = 1.4 nM T46828 CD6IC3 46231845 Ki = 7.5 nM T46828 C38WBY 46231846 Ki = 3.3 nM T46828 C0A7GW 46231847 Ki = 7.4 nM T46828 CVT82S 46231848 Ki = 26.9 nM T46828 C9W1US 46231924 Ki = 22 nM T46828 CL7WX9 46231925 Ki = 10 nM T46828 CVG26Z 46231926 Ki = 2.5 nM T46828 CKJ09A 46231927 Ki = 2.1 nM T46828 C2BX8U 46231994 Ki = 3.4 nM T46828 C7FD2G 46231995 Ki = 4.7 nM T46828 CYV52A 46232066 Ki = 6.2 nM T46828 C03LTM 46869265 Ki = 2800 nM T46828 C2LZJ0 49783209 Ki = 972 nM T46828 C57SMG 49783415 Ki > 10000 nM T46828 C0TG6I 49783419 Ki > 10000 nM T46828 C2RY0J 50878551 Ki > 10000 nM T46828 C1W6TV 50898777 Ki > 10000 nM T46828 CXMZ73 50898778 Ki > 10000 nM T46828 CE4KP1 51050257 Ki > 10000 nM T46828 C19ZKQ 52946556 Ki = 1.5 nM T46828 CPA2G4 52951481 Ki > 10000 nM T46828 CYP0I3 52951482 Ki > 10000 nM T46828 CSX14G 53321869 Ki > 10000 nM T46828 C32YWL 53324045 Ki = 121 nM T46828 CRQF15 53325242 Ki = 529 nM T46828 CLZ09P 53359025 Ki > 10000 nM T46828 CG24AT 53381002 Ki > 10000 nM T46828 CQ3AR0 56589560 Ki = 4.4 nM T46828 C4XGR3 56589561 Ki = 91.4 nM T46828 C9PHZ3 56594402 Ki = 657 nM T46828 C82IVX 56594533 Ki = 389 nM T46828 CT4J5C 56594534 Ki = 11.4 nM T46828 CH37LU 56663451 Ki > 10000 nM T46828 C1TC7Q 56963799 Ki > 10000 nM T46828 CV08WY 57391216 Ki = 1370 nM T46828 C07PMA 57391307 Ki = 2684 nM T46828 CWT20M 57393083 Ki = 3812 nM T46828 C3GW6L 57398351 Ki = 867 nM T46828 CZX05B 57401706 Ki = 3223 nM T46828 CYN38R 57401819 Ki = 1758 nM T46828 CO0XD2 57401820 Ki = 2808 nM T46828 CX0B5M 57403525 Ki = 414 nM T46828 C5RUP6 60167166 Ki > 10000 nM T46828 C34GMW 69599704 Ki > 10000 nM T46828 C9VZ8J 71450550 Ki > 10000 nM T46828 CE92DF 71528209 Ki = 5210 nM T46828 C31THM 72164180 Ki = 1743 nM T46828 C56VLM 72164181 Ki > 10000 nM T46828 CD8A9K 72164182 Ki = 1534 nM T46828 C4C0BH 72164183 Ki > 10000 nM T46828 CQU81Y 72164299 Ki > 10000 nM T46828 CF0H7K 72164300 Ki > 10000 nM T46828 C7WM5U 72164301 Ki > 10000 nM T46828 C4HO2U 72164302 Ki > 10000 nM T46828 CC65OA 73213195 Ki > 10000 nM T46828 CW83DK 73213196 Ki > 10000 nM T46828 CW8A0Y 73349359 Ki > 10000 nM T46828 CH2B4Y 73350932 Ki > 10000 nM T46828 C1NJ0R 73353884 Ki > 10000 nM T46828 CA4CP6 73355416 Ki > 10000 nM T46828 C81CIL 73355418 Ki > 10000 nM T46828 CN5V0R 73355421 Ki > 10000 nM T46828 C2E7QW 75201901 Ki = 4.8 nM T46828 CJG57Z 75202022 EC50 = 4.4 nM T46828 C8IDL3 75306277 Ki = 199.53 nM T46828 CZFW19 76314267 Ki = 17378.01 nM T46828 CIB40D 76321554 Ki = 3548.13 nM T46828 CS9F1X 76321556 Ki = 3467.37 nM T46828 C97LOB 76325150 Ki = 4570.88 nM T46828 CCR29U 76325152 Ki = 2454.71 nM T46828 CLP59V 76325156 Ki = 2754.23 nM T46828 C17YTI 76328715 Ki = 9700 nM T46828 CSW58A 76336021 Ki = 19498.45 nM T46828 C28RIZ 76518514 Ki > 10000 nM T46828 C8EWX5 85658088 Ki = 1613 nM T46828 CJ9K3T 86290953 EC50 > 10000 nM T46828 CM6X4U 86764103 EC50 = 12 nM T46828 C80SXV 90644057 Ki > 10000 nM T46828 CY8TP0 90644061 Ki = 2511.89 nM T46828 CKV24H 90644062 Ki = 1995.26 nM T46828 CW2ZC4 90644063 Ki = 3162.28 nM T46828 CLG60I 90644064 Ki > 10000 nM T46828 CKLN72 90644065 Ki > 10000 nM T46828 CDPE48 90644071 Ki = 1522 nM T46828 C35WTP 122177641 Ki = 24000 nM T46828 C8OS7B 122177642 Ki = 48000 nM T46828 CV2AT4 122177644 Ki = 21000 nM T46828 CB16GY 122177645 Ki = 700 nM T46828 CH9SX5 122180956 Ki = 3800 nM T46828 CCV9D5 122181326 Ki = 2800 nM T46828 C5D1NC 122181329 Ki = 2900 nM T46828 C05RGV 122181330 Ki = 7000 nM T46828 C3XGN0 122181333 Ki = 11000 nM T46828 CVJ3R4 122191605 Ki = 3600 nM T46828 C2J4ZX 122191607 Ki = 1300 nM T46828 C71KZQ 122205437 Ki = 3 nM T46828 C30ZRC 122205438 Ki = 1.9 nM T46828 CM57GR 126720252 Ki = 1070 nM T46828 C09YOS 127027905 Ki > 10000 nM T46828 CE9MN1 127028185 Ki > 10000 nM T46828 C9SC6E 127028505 Ki > 10000 nM T46828 CO53TS 127035828 Ki > 1000 nM T46828 CY7LP9 127035829 Ki > 1000 nM T46828 CR29BS 127035830 Ki > 1000 nM T46828 C50GOC 130442480 Ki = 82 nM T46828 CM04RF 130442572 Ki = 47 nM T46828 CAVB41 132584404 Ki > 10000 nM T46828 CBU81N 134149168 Ki > 10000 nM T46828 C5KE3N 135986088 Ki = 921 nM T46828 CN8BJ2 137632607 Ki > 20000 nM T46828 C3R2LO 137632761 Ki > 20000 nM T46828 C3PF9Z 137633454 Ki > 20000 nM T46828 CN1I7A 137634153 Ki > 20000 nM T46828 C6FRJ5 137634397 Ki > 15000 nM T46828 CPHI76 137635364 Ki = 3800 nM T46828 C8ZFQ6 137635685 Ki = 5800 nM T46828 CZ36LE 137636066 Ki = 15000 nM T46828 CAL1W4 137636298 Ki > 20000 nM T46828 CQ20FO 137636498 Ki = 3400 nM T46828 CZU6N5 137636581 Ki > 50000 nM T46828 C0YDQ5 137637428 Ki > 20000 nM T46828 C1HX3Z 137639304 Ki > 20000 nM T46828 CC16HE 137640152 Ki > 20000 nM T46828 CZP68A 137640189 Ki = 4200 nM T46828 C8IO0R 137640836 Ki > 20000 nM T46828 C6PT7L 137642033 Ki > 20000 nM T46828 CAC6W0 137643122 Ki > 20000 nM T46828 C71XIQ 137643132 Ki = 5700 nM T46828 C4PV8U 137645196 Ki > 20000 nM T46828 CNH95X 137645574 Ki = 9300 nM T46828 C3TP2G 137645830 Ki = 19000 nM T46828 CPI68E 137646281 Ki = 3016 nM T46828 CYH5U9 137647533 Ki > 20000 nM T46828 CW4T6D 137651322 Ki = 7700 nM T46828 CX30HQ 137653096 Ki > 20000 nM T46828 C4C6EV 137653986 Ki > 20000 nM T46828 COTX19 137654511 Ki > 20000 nM T46828 CF5Y2A 137654675 Ki = 13000 nM T46828 CLI4D8 137655029 Ki > 20000 nM T46828 CJAZ13 137655556 Ki > 20000 nM T46828 C6CA5H 137655594 Ki > 20000 nM T46828 CD16SQ 137655795 Ki = 16000 nM T46828 CE0Y7P 137657322 Ki > 20000 nM T46828 CRT86S 137657427 Ki > 20000 nM T46828 CH76FP 137657951 Ki > 20000 nM T46828 CP6US4 137660046 Ki = 16000 nM T46828 C5V4DQ 137660707 Ki > 20000 nM T46828 CL58XS 145967572 Ki = 286 nM T46828 C58WSL 145967904 Ki = 640 nM T46828 CB1FD8 145968810 Ki = 312 nM T46828 C48XNG 145969667 Ki = 101 nM T46828 CNZY06 145969934 Ki = 438 nM T46828 C61MSO 145970938 Ki = 605 nM T46828 C87MSW 145980271 Ki = 744 nM T46828 CNJH37 145986752 Ki = 623 nM T46828 CO4LK7 145988180 Ki = 143 nM T46828 CUGO10 145988693 Ki = 437 nM T46828 CC2G1V 146025727 Ki = 27 nM T46828 C6P3SR 153287553 Ki > 10000 nM T46828 CV9G7Z 153287572 Ki > 10000 nM T46828 CO85KL 153287574 Ki > 10000 nM T46828 CQ83KZ 155512662 Ki > 10000 nM T46828 CHXY56 155513802 Ki > 5000 nM T46828 CL5G9Q 155513837 Ki > 5000 nM T46828 CH34RK 155514798 Ki = 1204 nM T46828 CUE5J3 155515907 Ki > 5000 nM T46828 CUM2N4 155515982 Ki = 340 nM T46828 CV12SD 155516041 Ki > 5000 nM T46828 CJ98ZK 155516236 Ki > 5000 nM T46828 C9ZAW0 155517266 Ki = 5799 nM T46828 CUSA24 155519891 Ki > 10000 nM T46828 C8IYD1 155520455 Ki = 1995.3 nM T46828 C5DSE0 155520996 Ki = 1584.9 nM T46828 CV7IG5 155522663 Ki > 5000 nM T46828 C2H3JL 155523073 Ki = 1721 nM T46828 CQA76T 155523112 Ki > 5000 nM T46828 C3E9DJ 155523127 Ki > 5000 nM T46828 CVQ68Y 155523770 Ki = 2203 nM T46828 COH1Q5 155524191 Ki > 5000 nM T46828 CW7NT8 155524423 Ki = 3500 nM T46828 CQX27T 155525357 Ki > 5000 nM T46828 CW65KS 155525705 Ki = 1104 nM T46828 CKZ35G 155532475 Ki > 5000 nM T46828 C4LOR5 155532477 Ki > 5000 nM T46828 CQ12KS 155533996 Ki = 6109 nM T46828 C8AX5N 155534186 Ki = 7703 nM T46828 CHP2Z9 155535866 Ki = 9290 nM T46828 CB79ZW 155536080 Ki > 10000 nM T46828 CVFD68 155537516 Ki > 5000 nM T46828 C13CSU 155537907 Ki > 5000 nM T46828 C3DIY2 155539246 Ki = 926.1 nM T46828 CPV48W 155539557 Ki = 1000 nM T46828 CVK2M9 155543189 Ki = 8670 nM T46828 C4ANI0 155543691 Ki > 5000 nM T46828 C08FTE 155544239 Ki > 5000 nM T46828 C7MCZ0 155546478 Ki = 789 nM T46828 CN6I4P 155550431 Ki = 10532 nM T46828 C6N9PG 155550640 Ki > 5000 nM T46828 CG7NR9 155550756 Ki = 5580 nM T46828 C82QWR 155551173 Ki = 571 nM T46828 CX8JA1 155552185 Ki = 1000 nM T46828 CG70XQ 155552591 Ki = 8844 nM T46828 CB4F8Y 155552676 Ki = 1079.8 nM T46828 CD5LC6 155554006 Ki = 4227 nM T46828 C36SYJ 155558844 Ki > 5000 nM T46828 C7OZM6 155561446 Ki > 5000 nM T46828 CALB48 155561861 Ki > 10000 nM T46828 C2Z0HB 155562353 Ki = 2154.4 nM T46828 C0UN4V 155564747 Ki > 5000 nM T46828 CMH8I1 155565768 Ki = 8191 nM T46828 CK20WA 155566662 Ki > 5000 nM T46828 C6DPR8 155566974 Ki > 5000 nM T46828 C95RAP 155567835 Ki = 588.8 nM T46828 C5A6YM 155567869 Ki = 4018 nM T46828 CV24CW 155568676 Ki > 5000 nM T46828 C73ERT 155568786 Ki = 1847.9 nM T46828 C42JKO 155569198 Ki > 5000 nM T46828 C3N9VU 10251906 Ki > 500 nM T46828 CP9TR0 10324985 Ki > 10000 nM T46828 D00NQV 5041 Ki > 10000 nM T46828 D00SDJ 11237664 IC50 > 10000 nM T46828 D01ENR 2993172 Ki = 366 nM T46828 D04TWX 9794475 IC50 > 10000 nM T46828 D07RYR 44396235 Ki = 951 nM T46828 D09RPR 16737207 Ki > 10000 nM T46828 D0E1RX 11335419 Ki = 113 nM T46828 D0E3AL 56597938 Ki = 1100 nM T46828 D0F0IA 11301655 Ki > 8000 nM T46828 D0FF6S 16038374 IC50 > 10000 nM T46828 D0HH3R 11698643 Ki = 939 nM T46828 D0J1HP 10378389 Ki = 3715.35 nM T46828 D0L5MW 181743 Ki = 2397 nM T46828 D0L7OM 6917970 Ki = 4.4 nM T46828 D0L8PI 5018 IC50 = 0.56 nM T46828 D0LV7U 10667433 Ki = 330 nM T46828 D0R8UU 44396220 Ki = 43 nM T95913 D09XZB 123631 IC50 > 50000 nM T95913 D0B3HD 2519 IC50 = 1000000 nM T95913 D0E3SH 6918837 IC50 > 10000 nM T95913 D0E6XR 3062316 IC50 > 50000 nM T95913 D0F8RA 2153 IC50 = 800000 nM T95913 D0J5VR 11625818 IC50 = 60 nM T95913 D0K8KX 5280343 IC50 = 13790 nM T95913 D0R0MW 5329102 IC50 = 13000 nM T95913 D0RU0O 50905713 IC50 = 2 nM T95913 D0S5LD 135565596 IC50 = 0.7 nM T95913 D0W5HK 216239 IC50 > 50000 nM T95913 D01PGR 16123056 IC50 = 9 nM T95913 D01QSO 16654980 IC50 = 256 nM T95913 D03BHZ 52913813 IC50 = 675 nM T95913 D03EZE 25167777 IC50 = 0.61 nM T95913 D03FOP 68947304 IC50 = 850 nM T95913 D03IJO 11618268 IC50 = 3000 nM T95913 D03KAC 1893730 IC50 = 23 nM T95913 D03XAQ 49784945 IC50 = 36 nM T95913 D06GUA 49784002 IC50 = 6309.57 nM T95913 D07EHV 44814409 IC50 > 9100 nM T95913 D07HPJ 11476171 IC50 = 3200 nM T95913 D08QGT 17755052 Ki = 1.4 nM T95913 D0C3ZR 10427712 IC50 = 83 nM T95913 D0D8JB 44516953 IC50 = 6 nM T95913 D0E6UZ 54575456 IC50 = 311 nM T95913 D0I3LO 91933883 IC50 = 0.29 nM T95913 D0LG7X 86291103 IC50 = 33 nM T95913 D0O1LD 11647372 IC50 = 5 nM T95913 D0O6VZ 25254071 IC50 = 14 nM T95913 D0O8SJ 72950888 IC50 > 120 nM T95913 D0TU7B 58507717 IC50 = 708 nM T95913 D0U3DP 46912230 IC50 = 25 nM T95913 D0UP1Z 51001932 Ki = 0.97 nM T95913 D0VG0D 11977753 IC50 = 6 nM T95913 D0W7HE 56649450 IC50 = 250 nM T95913 D0X7IN 11978790 IC50 = 38 nM T95913 D0XD4I 118502708 IC50 = 1100 nM T95913 D0Y2NS 70798655 IC50 = 1900 nM T95913 D03BNU 59604787 IC50 > 5000 nM T95913 D0C9JZ 58111426 IC50 = 2297 nM T95913 D05HIJ 135565159 IC50 = 10000 nM T95913 D09SFV 3973 IC50 = 950 nM T95913 D0D0QA 44137675 IC50 = 1090 nM T95913 D0P1JI 312145 IC50 = 19 nM T95913 CX74ND 40237 IC50 = 380000 nM T95913 CEL9D8 79972 IC50 = 1498000 nM T95913 CNW59X 95001 IC50 = 53000 nM T95913 C3FRX9 131989 IC50 > 83300 nM T95913 C1MOD6 165595 IC50 = 2415000 nM T95913 CW1B9X 226105 IC50 = 1570000 nM T95913 C6KL2D 235602 IC50 = 992000 nM T95913 C4I2PT 244740 IC50 = 134000 nM T95913 C6ET7X 247414 IC50 = 5184000 nM T95913 CGC10Q 249363 IC50 = 2700 nM T95913 CQ7B2K 252311 IC50 = 187000 nM T95913 CBY29G 260801 IC50 = 105000 nM T95913 C1Y0JB 263480 IC50 = 324000 nM T95913 CTU12Q 267310 IC50 > 1600000 nM T95913 CJ43OR 270557 IC50 = 6074000 nM T95913 CV8DJ6 274101 IC50 = 241000 nM T95913 C2M5YF 275065 IC50 = 1460000 nM T95913 CEW10F 291727 IC50 = 234000 nM T95913 C1M3IR 309591 IC50 = 9157000 nM T95913 C6E4HJ 347279 IC50 = 5876000 nM T95913 CFW2K4 414938 IC50 = 2437000 nM T95913 COE1I6 426449 IC50 = 7333000 nM T95913 CK30NI 520127 IC50 > 1670000 nM T95913 CY3D4G 617191 IC50 = 16670 nM T95913 CS5O7B 622000 IC50 > 40000 nM T95913 CXC3V1 622262 IC50 = 1660 nM T95913 CU73NO 736009 IC50 > 83300 nM T95913 CZN6S9 743974 IC50 > 25118.86 nM T95913 C3P4OY 1093514 IC50 = 27950 nM T95913 C3KPX5 1270546 IC50 = 920 nM T95913 CP0QU1 1355022 IC50 = 3600 nM T95913 CWOQ49 1627922 IC50 = 10000 nM T95913 CAN89K 2762479 IC50 > 100000 nM T95913 C56YDF 2762944 IC50 > 100000 nM T95913 C8E3HY 2796894 IC50 = 5495.41 nM T95913 C09VKD 2816900 IC50 > 83300 nM T95913 C4RH3J 3106064 IC50 = 25000 nM T95913 C4PQ7T 3128427 IC50 = 5 nM T95913 C1O4KS 4416330 IC50 = 4200 nM T95913 CIN5F7 4904109 IC50 <= 10000 nM T95913 C1YJM9 4912089 IC50 > 83300 nM T95913 CE74CV 5059890 IC50 = 100000 nM T95913 C9N4MH 5765281 IC50 = 20000 nM T95913 CKX0F4 5806797 IC50 = 4300 nM T95913 C8CL1W 6053578 IC50 = 612000 nM T95913 CS26IV 6089668 IC50 = 3800 nM T95913 CGF7R0 6196488 IC50 = 20000 nM T95913 C2OZ0W 6484194 IC50 > 83300 nM T95913 CK2IR4 6852165 IC50 = 2030 nM T95913 CX18LU 9342140 IC50 = 1200 nM T95913 CE1Y8A 9815659 IC50 = 37000 nM T95913 CJ79RC 9879653 IC50 = 31 nM T95913 CC2Q6T 9925404 IC50 = 217800 nM T95913 CLT13A 10088066 IC50 = 4000 nM T95913 C9HWF6 10114067 IC50 = 3630 nM T95913 C57FPB 10115147 IC50 = 5450 nM T95913 CZ15SC 10125446 IC50 = 380 nM T95913 C02SQE 10141582 IC50 = 7620 nM T95913 CZ4D7S 10181657 IC50 = 145200 nM T95913 CF6Y2U 10202973 IC50 = 1820 nM T95913 C1RDW9 10203280 IC50 = 6170 nM T95913 CC82QV 10204538 IC50 = 137900 nM T95913 CO5VP9 10296641 IC50 = 2540 nM T95913 C7SFI1 10296883 IC50 > 10000 nM T95913 C7ZG0A 10296917 IC50 = 13070 nM T95913 CW7Q0R 10315189 IC50 = 18150 nM T95913 C32NQS 10357196 IC50 = 21 nM T95913 CC67FL 10383101 IC50 = 46000 nM T95913 C2VG4L 10455817 IC50 = 2.42 nM T95913 CAZT53 10475366 IC50 = 570 nM T95913 CL8YE3 11230964 IC50 = 6400 nM T95913 C8Y6IM 11234514 IC50 = 67 nM T95913 CK65NF 11418892 Ki = 3060 nM T95913 CL3Z4O 11419728 Ki = 20 nM T95913 CYBD21 11428504 IC50 = 100000 nM T95913 CHJ30L 11492951 IC50 = 250 nM T95913 C5E2PO 11500850 IC50 = 13500 nM T95913 CV8J3I 11514586 IC50 = 950 nM T95913 CTXF73 11515474 IC50 = 80 nM T95913 C0O4SQ 11522078 IC50 = 30 nM T95913 C7HMO6 11526786 IC50 = 8000 nM T95913 C15XPT 11529859 IC50 = 43 nM T95913 C5KV8L 11530037 IC50 = 530 nM T95913 CGK17J 11536358 IC50 = 110 nM T95913 C38YWS 11541283 IC50 = 6 nM T95913 C1VA4C 11543481 IC50 = 970 nM T95913 C4T8IQ 11550986 IC50 = 290 nM T95913 C63TOQ 11551198 IC50 = 39 nM T95913 CN2MS6 11562853 IC50 = 1258.93 nM T95913 C9JF1G 11565677 IC50 = 2600 nM T95913 CPXS32 11566902 IC50 = 56 nM T95913 CMVQ43 11576772 IC50 = 20 nM T95913 CUZP58 11580302 IC50 = 1000 nM T95913 CX92QM 11581007 IC50 = 29 nM T95913 CEHZ82 11599141 IC50 = 794.33 nM T95913 C6U0BN 11601532 IC50 > 10000 nM T95913 CL5F3Z 11601890 IC50 = 20 nM T95913 C58QVA 11601930 IC50 = 37 nM T95913 C1ZPM5 11630874 IC50 = 30 nM T95913 CLK3Y4 11638999 IC50 = 1000 nM T95913 CU2CK3 11644621 IC50 = 840 nM T95913 CQIX52 11645168 IC50 = 260 nM T95913 C08DUS 11645350 IC50 = 20000 nM T95913 CC64OJ 11652531 IC50 = 40 nM T95913 CP04JC 11666231 IC50 = 2.3 nM T95913 CK8T1S 11666950 IC50 = 29 nM T95913 CU0E8O 11690457 Ki > 4000 nM T95913 CLQ02O 11695207 IC50 = 20000 nM T95913 C3BT1M 11702204 IC50 = 20 nM T95913 CB0AP2 11705863 Ki > 4000 nM T95913 CY8C9P 11751126 IC50 = 382 nM T95913 CAJV97 11955205 IC50 = 21 nM T95913 CBR6D5 11955693 IC50 = 1860 nM T95913 C68SND 11955695 IC50 = 1873 nM T95913 C60DBM 11998444 IC50 > 40000 nM T95913 C5FTB0 11998445 IC50 = 6259 nM T95913 C68WMR 11998447 IC50 = 19790 nM T95913 CYL24B 11998448 IC50 = 16700 nM T95913 CNPI54 11998563 IC50 = 3506 nM T95913 C6AK0Y 11998564 IC50 = 1674 nM T95913 CMVA72 11998565 IC50 = 386 nM T95913 CJ3YP8 11998685 IC50 = 2076 nM T95913 CV8PB5 11998690 IC50 = 829 nM T95913 CB9T1H 11998803 IC50 = 49 nM T95913 C59SKD 11999032 IC50 = 31 nM T95913 CT58GS 12171624 IC50 = 333.96 nM T95913 C0RF3U 14501859 IC50 = 773000 nM T95913 CY7A0T 14638904 IC50 = 10900 nM T95913 CW2XK6 16050925 IC50 = 390 nM T95913 CW5FD8 16081736 IC50 = 16060 nM T95913 C2IF3P 16678352 IC50 > 30000 nM T95913 C3IO1C 16679060 IC50 > 30000 nM T95913 CV9US5 16736978 IC50 > 30000 nM T95913 C72THB 16739368 IC50 = 250 nM T95913 CF6JS9 16757570 IC50 = 54 nM T95913 CB19TH 16757576 IC50 = 10000 nM T95913 C9BJ7Q 16757577 IC50 = 660 nM T95913 C9DM4T 16757578 IC50 = 230 nM T95913 C1NZC7 16757579 IC50 > 10000 nM T95913 CY0S6G 17751063 IC50 = 127 nM T95913 CTP62W 17755300 IC50 = 9000 nM T95913 CQYN41 17755304 IC50 = 3000 nM T95913 C1G7NC 17755392 IC50 = 32700 nM T95913 CI87FV 17755495 IC50 = 17000 nM T95913 CI71OB 17755611 IC50 = 51000 nM T95913 C9W7ID 17755613 IC50 = 12.6 nM T95913 C1SN9M 17756679 IC50 >= 100000 nM T95913 CJAM62 18452190 IC50 = 11.2 nM T95913 C48LCH 18452193 IC50 = 4.27 nM T95913 CVH65S 18452195 IC50 = 2.66 nM T95913 C31KPH 18452198 IC50 = 4.76 nM T95913 CPSJ85 18452200 IC50 = 6.57 nM T95913 C14WMZ 18452237 IC50 = 2.59 nM T95913 CQ89PW 18452323 IC50 = 7.16 nM T95913 C1O3CJ 18452350 IC50 = 23 nM T95913 CXFA80 18452409 IC50 = 37.3 nM T95913 C9Q0EK 18452424 IC50 = 27.5 nM T95913 C5WV4J 18452430 IC50 = 103.4 nM T95913 CVDL81 22036885 IC50 = 6 nM T95913 C61ZGT 22135435 IC50 > 50118.72 nM T95913 CC5QS1 22263527 IC50 = 10890 nM T95913 CP05ZB 22346757 IC50 = 50000 nM T95913 C1F2TM 23582995 IC50 = 1500 nM T95913 CEYL29 23585510 Ki = 88 nM T95913 CR08WX 23586742 IC50 = 7260 nM T95913 CBL37C 23642173 Ki = 1020 nM T95913 C8J1SI 23642272 IC50 = 5285 nM T95913 C59CTR 23652981 IC50 = 97 nM T95913 C29SFI 24768579 IC50 = 829 nM T95913 C3M1OC 24802861 IC50 = 230 nM T95913 CP4G9Z 24855584 Ki = 120 nM T95913 CJV7D9 24855887 IC50 = 50 nM T95913 CM9C0R 24866805 IC50 = 6800 nM T95913 CB79YC 24905143 IC50 = 1500 nM T95913 C2DC9J 24905144 IC50 = 570 nM T95913 CN6V8Z 24905145 IC50 = 100 nM T95913 CSB7P5 24905148 IC50 = 2400 nM T95913 CGSF21 24905149 IC50 = 200 nM T95913 CVDG02 24905150 IC50 = 1800 nM T95913 CWH6C5 24905152 IC50 = 43 nM T95913 C0HE2Q 24905153 IC50 = 72 nM T95913 C7QSC9 24905154 IC50 = 990 nM T95913 CO9D0K 24905155 IC50 = 860 nM T95913 C5W9UR 24905157 IC50 = 1400 nM T95913 CC1DA3 24905158 IC50 = 940 nM T95913 COW79F 24905159 IC50 = 680 nM T95913 CFPA53 24905160 IC50 = 2400 nM T95913 C2O0JX 24905161 IC50 = 7200 nM T95913 CA72BE 24905162 IC50 = 900 nM T95913 CQN6X9 24905163 IC50 = 2400 nM T95913 CD4O1F 24905165 IC50 = 5900 nM T95913 CKL48T 24905166 IC50 = 10000 nM T95913 C76VYL 24905167 IC50 = 1300 nM T95913 C7K5PU 24905168 IC50 = 1400 nM T95913 CZ57ID 24905169 IC50 = 1100 nM T95913 C2DHX9 24905170 IC50 = 2300 nM T95913 CSB96E 24905171 IC50 = 100000 nM T95913 CWZ0R2 24905172 IC50 = 1100 nM T95913 CY3B6M 24905175 IC50 = 551 nM T95913 CW7UA3 24905176 IC50 = 821 nM T95913 CW1V0H 24905177 IC50 = 100000 nM T95913 CO6Y0L 24905178 IC50 = 100000 nM T95913 C60NQW 24905179 IC50 = 8020 nM T95913 C4MO8B 24905180 IC50 = 1470 nM T95913 COJI47 24905181 IC50 = 1210 nM T95913 CS0B2C 24905182 IC50 = 640 nM T95913 C1H4BT 24905183 IC50 = 271 nM T95913 C4WHK9 24905184 IC50 = 4250 nM T95913 C7Q4MZ 24905185 IC50 = 799 nM T95913 CS4IP1 24905186 IC50 = 270 nM T95913 C69QWO 24905187 IC50 = 873 nM T95913 C85ANB 24905188 IC50 = 123 nM T95913 CNHD75 24905189 IC50 = 87 nM T95913 C9JUO2 24905190 IC50 = 1022 nM T95913 CPR03K 24905191 IC50 = 1140 nM T95913 CTAG19 24905193 IC50 = 435 nM T95913 C7VJM5 24905194 IC50 = 430 nM T95913 CEP1L3 24905195 IC50 = 347 nM T95913 CP68ZD 24905196 IC50 = 239 nM T95913 C8Z0RJ 24905197 IC50 = 381 nM T95913 CN9RT0 24905198 IC50 = 100000 nM T95913 CHI78P 24905200 IC50 = 2700 nM T95913 CO6PE8 24905201 IC50 = 2000 nM T95913 CZ63HS 24905202 IC50 = 1300 nM T95913 C2X0FC 24905203 IC50 = 330 nM T95913 C0WCE3 24905204 IC50 = 220 nM T95913 CNK50B 24905205 IC50 = 590 nM T95913 C12DPB 24905206 IC50 = 830 nM T95913 C8N0RH 24905207 IC50 = 2700 nM T95913 CYA5G2 24905208 IC50 = 461 nM T95913 CDV2B4 24905209 IC50 = 1800 nM T95913 CEFK68 24905210 IC50 = 640 nM T95913 CUFP12 24905211 IC50 = 1300 nM T95913 C0JG8L 24905212 IC50 = 1500 nM T95913 CP47MK 24905213 IC50 = 15000 nM T95913 CB61QC 24905214 IC50 = 3000 nM T95913 CQ13ZI 24905215 IC50 = 100000 nM T95913 C6VI8F 24905216 IC50 = 184 nM T95913 CXNH25 24905217 IC50 = 167 nM T95913 C2PN9S 24905218 IC50 = 95 nM T95913 C9O2AL 24905219 IC50 = 228 nM T95913 CIT7U8 24905220 IC50 = 100000 nM T95913 CMD26S 24905221 IC50 = 627 nM T95913 C4R8WC 24905222 IC50 = 31000 nM T95913 C47SHA 24905223 IC50 = 113 nM T95913 C1DY2R 24905224 IC50 = 90 nM T95913 CS0XF9 24905225 IC50 = 100000 nM T95913 CG5VX2 24905226 IC50 = 100000 nM T95913 C57QEO 24905227 IC50 = 100000 nM T95913 C7CG5E 24905228 IC50 = 586 nM T95913 CHP5D1 24905229 IC50 = 3000 nM T95913 CXP09S 24905230 IC50 = 60 nM T95913 CY7XG1 24905231 IC50 = 7300 nM T95913 C7JFQ2 24905232 IC50 = 242 nM T95913 C2JM1P 24905233 IC50 = 6900 nM T95913 CC3BF0 24905234 IC50 = 3000 nM T95913 CE57FI 24905235 IC50 = 4200 nM T95913 CUP20O 24905236 IC50 = 3500 nM T95913 CLC6Q2 24905237 IC50 = 6200 nM T95913 C9M1GI 24905238 IC50 = 2400 nM T95913 CVD72F 24905239 IC50 = 101 nM T95913 CK38IZ 24905240 IC50 = 28 nM T95913 CO2V5E 24905241 IC50 = 22000 nM T95913 CZBA19 24905244 IC50 = 625 nM T95913 CQ8OI1 24905246 IC50 = 100000 nM T95913 C5URC6 24905247 IC50 = 4000 nM T95913 C03SVO 24905250 IC50 = 7700 nM T95913 CIF2J5 24905251 IC50 = 700 nM T95913 CPTE58 24905252 IC50 = 1450 nM T95913 CX1JB8 24905253 IC50 = 2400 nM T95913 COZ3H7 24905254 IC50 = 25000 nM T95913 CDT1H9 24905255 IC50 = 15000 nM T95913 C54QKA 24905256 IC50 = 1700 nM T95913 CRU3P2 24905257 IC50 = 100000 nM T95913 C9U0JA 24905259 IC50 = 11000 nM T95913 CO4YS7 24905260 IC50 = 9600 nM T95913 CEG0B5 24905261 IC50 = 100000 nM T95913 C9VE5F 24905262 IC50 = 100000 nM T95913 C3I4HK 24905264 IC50 = 20000 nM T95913 C0VMI6 24905265 IC50 = 100000 nM T95913 CWE3V0 24905267 IC50 = 100000 nM T95913 CH4T3A 24905268 IC50 = 50000 nM T95913 C6QDN7 24905271 IC50 = 3600 nM T95913 C6XHJ7 24905272 IC50 = 4500 nM T95913 CTB9A3 24905273 IC50 = 17000 nM T95913 C0NB1Q 24905274 IC50 = 6300 nM T95913 C9KQ0L 24905275 IC50 = 5100 nM T95913 C9O8QZ 24905277 IC50 = 4000 nM T95913 CP50RD 24905280 IC50 = 209 nM T95913 CG13ZM 24905281 IC50 = 735 nM T95913 CF0S6X 24905282 IC50 = 5160 nM T95913 C5HBL0 24905284 IC50 = 3340 nM T95913 C2Z5DN 24905285 IC50 = 852 nM T95913 CL6GH8 24905286 IC50 = 523 nM T95913 CKYO98 24905287 IC50 = 435 nM T95913 CRNQ65 24905288 IC50 = 340 nM T95913 COD7I5 24905289 IC50 = 772 nM T95913 C4LP7E 24905290 IC50 = 550 nM T95913 CE9JC2 24905291 IC50 = 200 nM T95913 C2GI1R 24905292 IC50 = 909 nM T95913 CHW8C4 24905293 IC50 = 355 nM T95913 CQF0H1 24905294 IC50 = 120 nM T95913 CNO7X0 24905295 IC50 = 140 nM T95913 C5WRG7 24905296 IC50 = 116 nM T95913 CQ1S0U 24905297 IC50 = 311 nM T95913 C4UES7 24905298 IC50 = 353 nM T95913 CMS69P 24905299 IC50 = 12500 nM T95913 CC0U5M 24905300 IC50 = 147 nM T95913 CW7X6S 24905301 IC50 = 16400 nM T95913 C97IQV 24905302 IC50 = 257 nM T95913 CSJ47V 24905303 IC50 = 1530 nM T95913 CPN74C 24905304 IC50 = 1820 nM T95913 C5CS3N 24905305 IC50 = 1390 nM T95913 CK4XE9 24905307 IC50 = 1070 nM T95913 CTU6Z3 24905308 IC50 = 100000 nM T95913 C9SQX1 24905309 IC50 = 780 nM T95913 CM75JP 24905310 IC50 = 1190 nM T95913 C9Q2BJ 24905311 IC50 = 1270 nM T95913 C9VUA1 24905312 IC50 = 366 nM T95913 CU3RS1 24905313 IC50 = 460 nM T95913 CYG3H2 24905314 IC50 = 633 nM T95913 CV5Q7O 24905315 IC50 = 283 nM T95913 C8SA3O 24905316 IC50 = 113 nM T95913 CI5MN3 24905317 IC50 = 58 nM T95913 CJ1P7K 24905318 IC50 = 43 nM T95913 C1T6YQ 24905319 IC50 = 554 nM T95913 CAU86X 24905320 IC50 = 342 nM T95913 C54ISY 24905321 IC50 = 808 nM T95913 C2GE5I 24905322 IC50 = 637 nM T95913 C8D6YK 24905323 IC50 = 606 nM T95913 C5NZH9 24905324 IC50 = 80 nM T95913 C9D6JR 24905325 IC50 = 1070 nM T95913 CLZT41 24905326 IC50 = 293 nM T95913 CW8FD3 24905327 IC50 = 808 nM T95913 CHB7A2 24905328 IC50 = 502 nM T95913 CA8EI3 24905329 IC50 = 448 nM T95913 CCQ0O7 24905330 IC50 = 1080 nM T95913 CJ81AS 24905331 IC50 = 39 nM T95913 C8PW4H 24905332 IC50 = 44 nM T95913 C2Y5TF 24905333 IC50 = 54 nM T95913 CH9FL5 24905334 IC50 = 2300 nM T95913 C1S0PC 24905335 IC50 = 1900 nM T95913 C8N9MV 24905336 IC50 = 7900 nM T95913 C9E8BJ 24905338 IC50 = 4000 nM T95913 CKZ80E 24905342 IC50 = 340 nM T95913 CO8SH1 24905343 IC50 = 200 nM T95913 C7IZL6 24905344 IC50 = 890 nM T95913 CLD3X6 24936051 IC50 = 47 nM T95913 C43VSW 24936353 IC50 = 501.19 nM T95913 C98MEW 24946175 IC50 = 6.7 nM T95913 CC7H3U 24946706 IC50 = 5.2 nM T95913 C78NJE 24955795 IC50 = 3130 nM T95913 C8P6NT 24956158 IC50 = 854 nM T95913 CJI29P 24956159 IC50 = 6654 nM T95913 C6C4RH 24993871 IC50 = 19 nM T95913 CL0TI6 24993895 IC50 = 6165.95 nM T95913 CS3Q8B 24995659 Ki > 4000 nM T95913 C8W3FZ 25023762 IC50 = 77.7 nM T95913 CZ9WE5 25023763 IC50 = 29.5 nM T95913 C3RL8W 25023764 IC50 = 36.1 nM T95913 CI6M9D 25023765 IC50 = 43.7 nM T95913 CF76VL 25023766 IC50 = 2.79 nM T95913 CC1KV3 25023767 IC50 = 2.34 nM T95913 CX7HP1 25023768 IC50 = 18.4 nM T95913 CEO7L0 25023769 IC50 = 33.2 nM T95913 CPA38V 25023770 IC50 = 1.92 nM T95913 C6QML7 25023771 IC50 = 4.28 nM T95913 C3VI4L 25023772 IC50 = 4.96 nM T95913 C6IOR9 25023773 IC50 = 4.84 nM T95913 CEW91Q 25032963 IC50 = 20 nM T95913 CY50OT 25052783 IC50 = 78 nM T95913 CHR51O 25057242 IC50 = 2600 nM T95913 CTM16Y 25069911 IC50 = 7909 nM T95913 CVI2S5 25070227 IC50 = 7582 nM T95913 CNL4Y2 25070228 IC50 = 11000 nM T95913 CSDN18 25070229 IC50 = 7907 nM T95913 CK92QL 25070230 IC50 = 10322 nM T95913 CKZ7X2 25070231 IC50 = 5830 nM T95913 C0T4NK 25070551 IC50 = 683 nM T95913 C1UKQ4 25070552 IC50 = 1378 nM T95913 CZRA03 25070553 IC50 = 2378 nM T95913 CO20FT 25070554 IC50 = 10000 nM T95913 CL4B5Z 25070555 IC50 = 1650 nM T95913 C7U0SC 25070882 IC50 = 1134 nM T95913 CCN36H 25071204 IC50 = 44 nM T95913 CQ7P4X 25071206 IC50 = 119 nM T95913 C14SFA 25071208 IC50 = 204 nM T95913 CNCJ40 25071516 IC50 = 61 nM T95913 CXWO13 25071518 IC50 = 776 nM T95913 CBH13R 25071519 IC50 = 1102 nM T95913 CJM7O0 25071520 IC50 = 594 nM T95913 C68PFD 25073081 IC50 = 583 nM T95913 CBJ20X 25073385 IC50 = 306 nM T95913 CZN7W0 25073388 IC50 = 368 nM T95913 CD69RK 25097993 IC50 = 33 nM T95913 CLP07J 25110819 IC50 > 10000 nM T95913 CVM89J 25128663 IC50 = 79.43 nM T95913 C4HRL9 25128667 IC50 = 39.81 nM T95913 C4SWT5 25128668 IC50 = 158.49 nM T95913 CIO6A4 25129024 IC50 = 630.96 nM T95913 CLS7P0 25129381 IC50 = 1995.26 nM T95913 C9R2EA 25129383 IC50 = 3981.07 nM T95913 C4YZL9 25129386 IC50 = 316.23 nM T95913 CDO9Q0 25129729 IC50 = 3981.07 nM T95913 CX86YV 25129734 IC50 = 398.11 nM T95913 CA2K4U 25130429 IC50 = 316.23 nM T95913 C1J8KH 25132804 IC50 = 3981.07 nM T95913 CI04XW 25132806 IC50 = 1000 nM T95913 C5WC4L 25133141 IC50 = 251.19 nM T95913 CSH37X 25133142 IC50 = 63.1 nM T95913 CW3HN6 25133144 IC50 = 1584.89 nM T95913 C4LHV1 25165368 IC50 > 10000 nM T95913 C2CXH3 25165371 IC50 > 10000 nM T95913 CQWL59 25165372 IC50 > 10000 nM T95913 CL87JW 25165773 IC50 = 7000 nM T95913 CB89TL 25165774 IC50 > 10000 nM T95913 CFZI92 25165961 IC50 > 10000 nM T95913 CK2YI4 25168990 IC50 = 6309.57 nM T95913 CC1D8V 25172062 IC50 = 14 nM T95913 CPW2D9 25172477 IC50 = 11 nM T95913 CLW96O 25207689 IC50 = 15 nM T95913 CWP29U 25242324 IC50 = 16 nM T95913 C4V2EJ 25261231 IC50 = 148 nM T95913 C3IDN0 25266674 IC50 = 12589.25 nM T95913 CIXE02 28063903 IC50 = 915000 nM T95913 C2IM0O 39733146 IC50 = 2511.89 nM T95913 CO4PL8 42606076 IC50 > 100000 nM T95913 C20VGT 42606077 IC50 = 40000 nM T95913 C7N5EC 42606078 IC50 > 100000 nM T95913 CIF63E 42623219 IC50 = 100 nM T95913 C3DNM9 42623223 IC50 = 25.12 nM T95913 COR5I0 42623224 IC50 = 251.19 nM T95913 CX1DC2 42623385 IC50 = 6.31 nM T95913 CR6N3I 42623632 IC50 = 15.85 nM T95913 C4EM0W 42623869 IC50 = 630.96 nM T95913 C5TY9Q 42623950 IC50 = 158.49 nM T95913 C10RBA 42636535 IC50 = 8000 nM T95913 C8N6CY 44119296 IC50 = 156000 nM T95913 C3ROX1 44124863 Ki = 1.9 nM T95913 CI3K7H 44129042 IC50 = 7900 nM T95913 CIE0J3 44129043 IC50 > 10000 nM T95913 CUW85V 44129044 IC50 > 10000 nM T95913 C2B9DE 44129118 IC50 = 8300 nM T95913 C0R1PH 44129198 IC50 > 10000 nM T95913 C6LGD5 44129200 IC50 = 3000 nM T95913 C03RLS 44129270 IC50 > 10000 nM T95913 CU4H1I 44129274 IC50 > 10000 nM T95913 C79QOC 44129275 IC50 = 6100 nM T95913 C0W3ZF 44129348 IC50 > 10000 nM T95913 CH6RO4 44129351 IC50 > 10000 nM T95913 CPAU59 44129353 IC50 > 10000 nM T95913 CN5O4I 44129429 IC50 = 2900 nM T95913 C3ZSV2 44129432 IC50 = 6300 nM T95913 CM5U2I 44137407 IC50 = 211 nM T95913 CQ82MS 44138035 IC50 = 23000 nM T95913 CZA3N9 44138128 IC50 = 34000 nM T95913 CF17OS 44180029 IC50 = 808 nM T95913 CHK8Z6 44180034 IC50 = 1170 nM T95913 CEJ5F7 44180035 IC50 = 9180 nM T95913 CQNT23 44180155 IC50 = 158 nM T95913 CIKM57 44180156 IC50 = 1310 nM T95913 CBP2T3 44180157 IC50 = 1090 nM T95913 C9CGB4 44180282 IC50 = 503 nM T95913 C2S5LC 44180395 IC50 = 410 nM T95913 C40NOQ 44180397 IC50 = 1080 nM T95913 CTB46H 44180398 IC50 = 547 nM T95913 CRS2G3 44180853 IC50 = 3945 nM T95913 C2VZX7 44181492 IC50 > 50000 nM T95913 C7SYM2 44181493 IC50 = 8780 nM T95913 CB8KF1 44181494 IC50 = 5460 nM T95913 C5AI8R 44181598 IC50 = 4220 nM T95913 CK03RW 44181599 IC50 = 2310 nM T95913 CXL61J 44181600 IC50 = 1570 nM T95913 C6TZK5 44181601 IC50 = 385 nM T95913 CCIV74 44181602 IC50 = 553 nM T95913 C36WUP 44181603 IC50 > 50000 nM T95913 CS2U7R 44181604 IC50 = 6300 nM T95913 CL6W0C 44181605 IC50 = 314 nM T95913 CFD41Z 44181718 IC50 = 7500 nM T95913 C2RB1P 44181719 IC50 = 5200 nM T95913 CMC75I 44181720 IC50 = 1390 nM T95913 CWTS93 44181721 IC50 = 667 nM T95913 CT1JL2 44181722 IC50 = 586 nM T95913 CE9HO1 44181723 IC50 = 5560 nM T95913 CFSB29 44181724 IC50 = 4990 nM T95913 CS0M9A 44187604 IC50 = 18.5 nM T95913 C0BRI9 44187779 IC50 = 37 nM T95913 CDA81B 44187783 IC50 = 25 nM T95913 C0LB8S 44187784 IC50 = 11.5 nM T95913 CCTO21 44187951 IC50 = 84.5 nM T95913 CVYS60 44187952 IC50 = 12 nM T95913 C8X3UZ 44187955 IC50 = 9 nM T95913 CJU85Z 44188321 IC50 = 33 nM T95913 CHU02A 44188322 IC50 = 17.2 nM T95913 C69HQS 44188840 IC50 = 13.5 nM T95913 CD78AG 44188841 IC50 = 19.5 nM T95913 CY7EL1 44188842 IC50 = 21.5 nM T95913 C0SE1X 44188843 IC50 = 48.5 nM T95913 CG13ZF 44188844 IC50 = 24.8 nM T95913 CR0BF9 44189010 IC50 = 78 nM T95913 C71NFL 44189011 IC50 = 69 nM T95913 C39ABJ 44189192 IC50 = 17.5 nM T95913 CK73NR 44219749 IC50 = 6315 nM T95913 CZ3L7W 44233390 IC50 = 1697 nM T95913 CA7R1U 44233391 IC50 = 1772 nM T95913 CU2F9E 44413107 IC50 = 29 nM T95913 C9SK8P 44413114 IC50 = 200 nM T95913 C9ZML1 44454396 IC50 = 117 nM T95913 CVG75D 44473371 IC50 = 8 nM T95913 C30NZA 44475985 IC50 = 69 nM T95913 CAT8F7 44475986 IC50 = 185 nM T95913 CSR73H 44475987 IC50 = 1300 nM T95913 CDAX92 44475988 IC50 = 113 nM T95913 CBH0S5 44475989 IC50 = 20000 nM T95913 CW5A7L 44475990 IC50 = 4 nM T95913 CLKU13 44481151 Ki = 39 nM T95913 CX3FK1 44513884 IC50 = 28.5 nM T95913 CL4RO5 44513885 IC50 = 34 nM T95913 C6RC9J 44513886 IC50 = 27 nM T95913 CGS7Q4 44513887 IC50 = 23 nM T95913 CSVD32 44513888 IC50 = 438 nM T95913 CLN2M5 44514201 IC50 = 52.5 nM T95913 C2Y8ML 44514203 IC50 = 219.5 nM T95913 CA9H8D 44514205 IC50 = 528 nM T95913 C01ZJI 44514208 IC50 = 18 nM T95913 CZ8WK6 44514210 IC50 = 24.5 nM T95913 CI8H3K 44514481 IC50 = 814.5 nM T95913 C51SEJ 44515083 IC50 = 21.5 nM T95913 CXBV98 44515084 IC50 = 14.5 nM T95913 C73HNB 44515696 IC50 = 85 nM T95913 CB7XW5 44516307 IC50 = 48.5 nM T95913 C4W5EM 44516309 IC50 = 9 nM T95913 C8VAU1 44516310 IC50 = 20 nM T95913 C8I1ZB 44516311 IC50 = 9 nM T95913 CSJ95V 44516635 IC50 = 10 nM T95913 CV6Z0N 44516636 IC50 = 10 nM T95913 CB3MV8 44517288 IC50 = 49.5 nM T95913 CDEQ97 44520808 IC50 = 993 nM T95913 CB4RN0 44520812 IC50 = 2367 nM T95913 CFC65B 44539960 IC50 <= 1000 nM T95913 C03IGD 44540030 IC50 = 7943.28 nM T95913 C5LWU1 44540126 IC50 = 7943.28 nM T95913 CYD4Z8 44540130 IC50 = 50.12 nM T95913 CAT2R7 44540316 IC50 = 15848.93 nM T95913 C36NRP 44540403 IC50 <= 1000 nM T95913 C2T9GC 44540407 IC50 = 6309.57 nM T95913 CQ4PE7 44540492 IC50 > 25118.86 nM T95913 C6HC3L 44548482 IC50 = 72.5 nM T95913 CH3L9P 44551660 IC50 > 1000 nM T95913 CYMD49 44552663 IC50 = 1358 nM T95913 C6B7LH 44552664 IC50 = 473 nM T95913 C3QZX0 44552666 IC50 = 283 nM T95913 C64OQC 44552667 IC50 = 155 nM T95913 C7LG6Q 44552844 IC50 = 404 nM T95913 C9T2CZ 44552845 IC50 = 76 nM T95913 CXLD75 44552846 IC50 = 109 nM T95913 CALT95 44554240 IC50 = 2781 nM T95913 CVDA08 44554755 IC50 = 1458 nM T95913 C25EGX 44554909 IC50 = 1820 nM T95913 CR4J0X 44554913 IC50 = 1625 nM T95913 CWV2T9 44554915 IC50 = 402 nM T95913 CCW12H 44555222 IC50 = 269 nM T95913 CTM8S9 44555225 IC50 = 2419 nM T95913 C7PSO6 44555226 IC50 = 646 nM T95913 C3VRO9 44557921 IC50 = 12.59 nM T95913 CRE61W 44577592 IC50 = 258 nM T95913 CH63GM 44577593 IC50 = 113 nM T95913 CA8MV5 44577594 IC50 = 321 nM T95913 C9IXW8 44577638 IC50 = 159 nM T95913 C8A5RT 44577639 IC50 = 28 nM T95913 CNP02V 44577640 IC50 = 73 nM T95913 CT6GN5 44577641 IC50 = 189 nM T95913 CIQR97 44577850 IC50 = 959 nM T95913 CCG8P9 44577851 IC50 = 16840 nM T95913 CLBA40 44577853 IC50 = 357 nM T95913 COU6V7 44577854 IC50 = 531 nM T95913 C8M5FY 44577914 IC50 = 318 nM T95913 C3MGZ9 44577915 IC50 > 20000 nM T95913 CGO09K 44577916 IC50 = 80 nM T95913 CRJ3B7 44577917 IC50 = 210 nM T95913 CTR89C 44577918 IC50 > 20000 nM T95913 CO05YG 44577919 IC50 = 163 nM T95913 CT70WA 44577920 IC50 = 77 nM T95913 C5KXS4 44577921 IC50 = 145 nM T95913 CZ2HI5 44577922 IC50 = 107 nM T95913 CGTU34 44577950 IC50 = 819 nM T95913 CQC50R 44577951 IC50 = 52 nM T95913 C8ZTW2 44577952 IC50 = 440 nM T95913 CIL93G 44577953 IC50 = 617 nM T95913 C8NB5H 44578037 IC50 > 40000 nM T95913 CX9TO2 44578038 IC50 = 35730 nM T95913 C7AHR4 44578039 IC50 > 50000 nM T95913 C13LGI 44578040 IC50 > 50000 nM T95913 CNZ06H 44578074 IC50 > 50000 nM T95913 C41TYA 44578108 IC50 = 63 nM T95913 C2W3SQ 44578109 IC50 = 223 nM T95913 CYM69I 44580064 IC50 = 51 nM T95913 CV09JM 44580065 IC50 = 34 nM T95913 CF37TO 44580066 IC50 = 35 nM T95913 CA0BU6 44580067 IC50 = 203 nM T95913 COQ85J 44580235 IC50 = 24 nM T95913 CD4ER0 44580236 IC50 = 20 nM T95913 CHVQ28 44580237 IC50 = 34 nM T95913 C8N2AF 44580238 IC50 = 767 nM T95913 C40LVX 44580274 IC50 = 1288 nM T95913 CO9LD8 44580275 IC50 = 138 nM T95913 C5QWG4 44580276 IC50 = 222 nM T95913 CFZS45 44580277 IC50 = 174 nM T95913 CQ4CR6 44580635 IC50 = 201 nM T95913 CJHK57 44580636 IC50 = 257 nM T95913 CC6M2E 44580684 IC50 = 70 nM T95913 CA3KP5 44580685 IC50 = 180 nM T95913 C40VHS 44580686 IC50 = 52 nM T95913 CXV92J 44580687 IC50 = 767 nM T95913 CG3PH2 44580721 IC50 = 327 nM T95913 CIO46B 44580722 IC50 = 48 nM T95913 CNLS71 44580723 IC50 = 35 nM T95913 C1N0MF 44580724 IC50 = 18 nM T95913 CAHQ76 44580766 IC50 = 131 nM T95913 C2XN6B 44580767 IC50 = 51 nM T95913 CC36YN 44580768 IC50 = 70 nM T95913 CZ56FY 44580769 IC50 = 46 nM T95913 CL8S0Y 44592136 IC50 >= 50000 nM T95913 C9E6JV 44592170 IC50 = 10000 nM T95913 C8DUA1 44592171 IC50 < 10000 nM T95913 CY8VU1 44592172 IC50 < 10000 nM T95913 C56TOC 44592173 IC50 < 10000 nM T95913 CGP6M7 44592216 IC50 >= 100000 nM T95913 CS38JL 44592217 IC50 = 100000 nM T95913 CJ1FW0 44592218 IC50 > 100000 nM T95913 C70VRG 44592219 IC50 > 100000 nM T95913 CW5RQ0 44592258 IC50 > 100000 nM T95913 CVB1I3 44592259 IC50 > 100000 nM T95913 CV9MY8 44592260 IC50 > 100000 nM T95913 CA65CE 44592261 IC50 > 100000 nM T95913 CEHY48 44592262 IC50 > 100000 nM T95913 C09OLK 44592299 IC50 = 42000 nM T95913 CJM35R 44592300 IC50 > 100000 nM T95913 C54DKW 44592302 IC50 = 42000 nM T95913 CJX76V 44592338 IC50 > 100000 nM T95913 CNY53M 44592339 IC50 > 100000 nM T95913 CXPK04 44592340 IC50 > 100000 nM T95913 C0L2HO 44593630 IC50 = 107 nM T95913 C2NQ6Z 44593631 IC50 = 22 nM T95913 CHKQ45 44593990 IC50 > 10000 nM T95913 CY3SV7 44596118 IC50 > 10000 nM T95913 C28QLM 44605035 IC50 = 6224 nM T95913 C75XHS 44605037 IC50 = 495 nM T95913 C3F4UX 44605249 IC50 = 1431 nM T95913 CQ0FZ7 44605426 IC50 = 3765 nM T95913 CC7G2L 44605427 IC50 = 3554 nM T95913 CDLP04 44605428 IC50 = 409 nM T95913 CSKN09 44605429 IC50 = 2526 nM T95913 CA79QG 44605430 IC50 = 1290 nM T95913 CH6V9F 44608754 IC50 = 6.5 nM T95913 C0IY9N 44608757 IC50 = 16 nM T95913 C90ITS 44608915 IC50 = 8.1 nM T95913 CZH1P9 44609387 IC50 = 2.4 nM T95913 CNDX48 44609388 IC50 = 13 nM T95913 CE95RQ 44620964 IC50 = 15 nM T95913 CVYJ36 44620965 IC50 = 33 nM T95913 CA8BY7 44621440 IC50 = 31.62 nM T95913 C5M1FR 44621441 IC50 = 25.12 nM T95913 C5LD7E 44621442 IC50 = 7.943 nM T95913 CO4GT0 44621447 IC50 = 25.12 nM T95913 CUV26H 44621448 IC50 = 19.95 nM T95913 CV2MG9 44621449 IC50 = 19.95 nM T95913 C24IYW 44621451 IC50 = 39.81 nM T95913 C0F9YW 44621452 IC50 = 100 nM T95913 C0GRD8 44621454 IC50 = 79.43 nM T95913 C4YHJ0 44621456 IC50 = 19.95 nM T95913 C31VBF 44621458 IC50 = 15.85 nM T95913 CQD03G 44623048 Ki = 770 nM T95913 C54IUP 44818842 IC50 = 435 nM T95913 C16IMZ 44819024 IC50 = 49 nM T95913 CN38JF 44819199 IC50 = 48.5 nM T95913 CVW6L8 44819200 IC50 = 22 nM T95913 CZ7M6D 44819201 IC50 = 12.2 nM T95913 C7MU8J 44819203 IC50 = 12.3 nM T95913 C8FU0W 44819375 IC50 = 22 nM T95913 C4N8CK 44819376 IC50 = 25 nM T95913 CP6DB9 45265864 IC50 = 40 nM T95913 C5I1VH 45379222 IC50 = 789 nM T95913 CA4JZ8 45379223 IC50 = 65 nM T95913 CZ68MG 45488079 IC50 > 10000 nM T95913 CV1U7I 46180604 IC50 = 8.4 nM T95913 CED2B3 46180606 IC50 = 5100 nM T95913 CDV85O 46180663 IC50 = 1300 nM T95913 CZGB46 46180666 IC50 = 15 nM T95913 C61ZLI 46190736 IC50 = 265 nM T95913 C6H3GT 46196486 IC50 = 33 nM T95913 CAU17V 46202808 IC50 = 3.162 nM T95913 CDA3R9 46220225 IC50 = 8 nM T95913 CIJ5V9 46224766 IC50 = 223 nM T95913 CIPV59 46224808 IC50 = 640 nM T95913 CRQ5M4 46225259 IC50 = 10000 nM T95913 C65IPQ 46225280 IC50 = 133 nM T95913 C8A7QJ 46225281 IC50 = 341 nM T95913 CPL45H 46225307 IC50 = 6907 nM T95913 CTN8J2 46225308 IC50 = 8297 nM T95913 CL34IK 46227801 IC50 = 510 nM T95913 C6D2RL 46227820 IC50 = 975 nM T95913 CSIK15 46228569 IC50 = 7470 nM T95913 C94YRI 46853654 IC50 = 3.981 nM T95913 CZ3WS1 46861592 IC50 = 5 nM T95913 CRO8W0 46865423 IC50 = 25 nM T95913 C47VTS 46865424 IC50 = 11 nM T95913 CO3P0J 46866604 IC50 = 1256 nM T95913 CQ2Y1V 46866705 Ki = 0.111 nM T95913 C63RCG 46870269 IC50 = 2.512 nM T95913 CTQ25M 46871497 IC50 = 6.31 nM T95913 CXRI03 46872177 Ki = 0.048 nM T95913 CC0R5U 46872178 Ki = 0.017 nM T95913 C8SRB0 46872297 Ki = 0.157 nM T95913 C67QZY 46872298 Ki = 0.33 nM T95913 CQB16A 46872415 Ki = 0.003 nM T95913 C7V8RJ 46873664 Ki = 0.066 nM T95913 CJB8T7 46873665 Ki = 0.011 nM T95913 CU7Z9M 46873667 Ki = 0.013 nM T95913 C6MZ1J 46884121 IC50 = 6949 nM T95913 CLA40T 46885426 IC50 = 3628 nM T95913 CC8T1E 46885496 IC50 = 2220 nM T95913 CCS20H 46885565 IC50 = 10 nM T95913 CG47YP 46885566 IC50 = 587 nM T95913 C4R3XP 46885599 IC50 = 54 nM T95913 CV5MK6 46885601 IC50 = 976 nM T95913 C42WVO 46885648 IC50 = 322 nM T95913 C3HMQ2 46891474 IC50 = 2.4 nM T95913 CB6Z8P 46892208 IC50 = 6200 nM T95913 CZX46Y 46892342 IC50 = 110 nM T95913 C5FN6I 46892845 IC50 = 320 nM T95913 CQ32BN 46892970 IC50 = 8 nM T95913 COJA32 46892971 Ki = 69 nM T95913 C5QFB3 46893088 IC50 = 200 nM T95913 CS30AI 46893754 IC50 = 3600 nM T95913 CPO1N7 46927938 Ki = 179 nM T95913 CJ0VB4 46932297 IC50 = 430 nM T95913 CL84AF 46946248 Ki > 500 nM T95913 CF14PE 46947264 IC50 = 74 nM T95913 COE37N 49778924 IC50 = 790 nM T95913 C7ZK3D 49783923 IC50 = 316.23 nM T95913 CHX76J 49784892 Ki = 29 nM T95913 CA1H8S 49784893 Ki = 88 nM T95913 CP2QD0 49784894 Ki = 4 nM T95913 CTZG05 49784988 Ki = 45 nM T95913 CE9AC5 49785078 Ki = 23 nM T95913 CG2IO7 49785079 Ki = 12 nM T95913 C8EYN4 49785083 Ki = 17 nM T95913 CBNZ47 49785166 Ki = 136 nM T95913 CZI34V 49785167 Ki = 330 nM T95913 CJK65T 49785253 Ki = 51 nM T95913 CXK8F5 49785436 Ki = 2 nM T95913 CWL5C6 49785518 Ki = 6 nM T95913 C3NV0J 49785827 Ki = 12 nM T95913 C0OZM2 49785828 Ki = 200 nM T95913 C1AR4G 49785829 Ki = 450 nM T95913 C39HAK 49785832 Ki = 12 nM T95913 C90JBE 49834576 IC50 > 10000 nM T95913 C5UR4A 49843944 IC50 = 720 nM T95913 CS40YB 49853846 IC50 = 230 nM T95913 C7PER0 49853953 IC50 = 660 nM T95913 CU9A8O 49854022 IC50 > 10000 nM T95913 C51QVH 49854023 IC50 = 10000 nM T95913 CM4HQ2 49854024 IC50 > 10000 nM T95913 C1LBX3 49854049 IC50 = 430 nM T95913 CVC2H6 49854052 IC50 = 290 nM T95913 CC2X9N 49854121 IC50 > 10000 nM T95913 CAJ58E 49854156 IC50 = 180 nM T95913 CAU39Y 49854158 IC50 = 200 nM T95913 CPK6X3 49854360 IC50 = 1400 nM T95913 CBVT70 49854361 IC50 = 4000 nM T95913 CQ1TZ6 49854365 IC50 = 1100 nM T95913 CJ5I9X 49854461 IC50 = 330 nM T95913 CDXQ69 49854462 IC50 = 8000 nM T95913 C0ORZ9 49854466 IC50 = 200 nM T95913 CY14XF 49854572 IC50 = 1200 nM T95913 CEC10T 49854573 IC50 = 15 nM T95913 C39KQW 49854679 IC50 = 200 nM T95913 C8VDR2 49854680 IC50 = 160 nM T95913 CN2V8R 49854681 IC50 = 990 nM T95913 CSN96A 49855001 IC50 = 230 nM T95913 CALY90 49855192 IC50 = 5000 nM T95913 CJPE20 49855193 IC50 = 2500 nM T95913 C1OM3I 49855237 IC50 = 17780 nM T95913 C26IQK 49857091 IC50 = 5300 nM T95913 CR0PN9 49857092 IC50 = 5700 nM T95913 CCJN26 49857093 IC50 = 1900 nM T95913 C3YG5L 49857275 IC50 > 10000 nM T95913 CHO65B 49857279 IC50 = 2640 nM T95913 C9HMY1 49857280 IC50 = 1800 nM T95913 CGW9L1 49857476 IC50 = 5150 nM T95913 CRD84P 49857479 IC50 = 1400 nM T95913 COF78C 49857678 IC50 > 10000 nM T95913 C4H7XG 49857865 IC50 = 2200 nM T95913 CY8MP7 49867926 IC50 = 9 nM T95913 CR0IA5 49871864 IC50 = 1100 nM T95913 C13WJZ 49872243 IC50 = 290 nM T95913 C5OY7B 49872246 IC50 = 146 nM T95913 C2KD5E 49872344 IC50 = 62 nM T95913 CV5BF3 49872645 IC50 = 634 nM T95913 CN97FO 49872646 IC50 = 22.5 nM T95913 CD6P5R 49872735 IC50 = 507 nM T95913 CL64NB 49872737 IC50 = 4650 nM T95913 CRNG04 49872831 IC50 = 11 nM T95913 CQC8B4 49872835 IC50 = 13 nM T95913 CPS3O1 49872924 IC50 = 120 nM T95913 CUBX74 49872925 IC50 = 19 nM T95913 CAW69U 49872927 IC50 = 220 nM T95913 CV1L4P 49873242 IC50 = 964 nM T95913 C5BA2V 49873243 IC50 = 3590 nM T95913 CSN45W 49873329 IC50 = 35.4 nM T95913 CLC2N7 50913517 IC50 = 20500 nM T95913 CJ4L8Y 50938829 Ki = 364 nM T95913 CJG65L 50939078 Ki = 509 nM T95913 CI8QM1 50939080 Ki = 28 nM T95913 CT0IP3 50939081 Ki = 90 nM T95913 C54EUL 50939212 Ki = 7340 nM T95913 CS7Z6U 50939338 Ki = 92 nM T95913 C2I9PS 50939992 IC50 = 18000 nM T95913 C9TUE4 50940108 IC50 = 1400 nM T95913 C2Q0GE 50990922 IC50 = 100 nM T95913 CKY3V1 50990924 Ki = 4.7 nM T95913 C5ZF9W 51003380 IC50 = 77000 nM T95913 CY36EH 51003592 IC50 = 398.11 nM T95913 CLB85F 51346892 IC50 = 740 nM T95913 C65ILG 51346893 IC50 = 44 nM T95913 CRJ5W8 51358113 IC50 = 5.67 nM T95913 CT91WR 52040626 IC50 = 371 nM T95913 CG7T4H 52913198 IC50 = 25 nM T95913 CD84MT 52913592 IC50 = 2200 nM T95913 C2TLG6 52913931 IC50 = 1800 nM T95913 CQ5GF2 52917084 Ki = 126 nM T95913 CAFR91 52917382 Ki = 361 nM T95913 C2DQK4 52917534 Ki = 50.1 nM T95913 C5ON6F 52919356 IC50 = 14 nM T95913 CM5BX0 52919492 IC50 = 68 nM T95913 CU1P2L 52940797 IC50 = 2010 nM T95913 CD62QJ 52940982 IC50 = 358 nM T95913 C43SVQ 52941322 IC50 = 189.5 nM T95913 CK59HM 52941479 IC50 = 150 nM T95913 C2KI6V 52942202 IC50 = 100000 nM T95913 CFRN73 52942850 IC50 = 122 nM T95913 C4D1KT 52942879 IC50 = 44 nM T95913 C4VCY0 52943258 IC50 = 16000 nM T95913 C1XEV2 52943394 IC50 = 2410 nM T95913 C73WTL 52943744 IC50 = 45.2 nM T95913 C6Q1AH 52943745 IC50 = 100 nM T95913 CHI0P6 52944356 IC50 = 100000 nM T95913 CWD27C 52945142 IC50 = 240 nM T95913 CWPC54 52945348 IC50 = 140 nM T95913 CXL53B 52945589 IC50 = 154 nM T95913 C4NLX7 52945630 IC50 = 723 nM T95913 CXD6T8 52945845 IC50 = 1200 nM T95913 CN8F0V 52946289 IC50 = 717 nM T95913 CMQY93 52946368 IC50 = 149 nM T95913 C5X9VO 52948007 IC50 = 290 nM T95913 C7ET6Z 52948010 IC50 = 1600 nM T95913 CW9Z1T 52949347 IC50 = 51 nM T95913 CV5B2C 52949497 IC50 = 25000 nM T95913 CB0KM5 52949869 IC50 = 98 nM T95913 CAJQ03 52950001 IC50 = 99 nM T95913 C5HQ2E 52950102 IC50 = 74 nM T95913 CH1Q5D 53234281 IC50 = 3 nM T95913 C45JKN 53234283 IC50 = 8.4 nM T95913 CVK28S 53235062 IC50 = 0.7 nM T95913 COW61E 53235216 IC50 = 1.5 nM T95913 CWE56X 53235217 IC50 = 3.7 nM T95913 CDXM59 53235451 IC50 = 55 nM T95913 CT8IN1 53242225 IC50 = 3200 nM T95913 C9NF0C 53302364 Ki = 42.4 nM T95913 C4J9WZ 53307606 IC50 = 5 nM T95913 C7ZH0D 53308041 IC50 = 1170 nM T95913 CRD3A9 53316967 IC50 = 340 nM T95913 C84YNK 53317325 IC50 > 83300 nM T95913 CS8DJ3 53318252 IC50 = 150 nM T95913 C58NQJ 53318614 IC50 = 55400 nM T95913 C10YUH 53318615 IC50 = 9700 nM T95913 C24GBF 53319075 IC50 = 15 nM T95913 CFJD70 53319932 IC50 = 70000 nM T95913 C3EJB1 53319933 IC50 = 9100 nM T95913 C2V7AX 53320017 IC50 = 380 nM T95913 CKGJ60 53320018 IC50 = 730 nM T95913 CJRM64 53322563 IC50 = 43500 nM T95913 CN92LK 53322732 IC50 = 9 nM T95913 CJZ29M 53325374 IC50 = 830 nM T95913 C1TE8J 53325515 IC50 = 7600 nM T95913 C6LAI9 53326166 IC50 = 960 nM T95913 CCU75P 53327266 Ki = 6 nM T95913 C1TWE6 53327269 Ki = 3 nM T95913 COSB47 53327579 Ki = 20 nM T95913 C62JOP 53327629 Ki = 4 nM T95913 CCX7M5 53353847 Ki = 20.7 nM T95913 C23HAU 53361718 IC50 = 7.7 nM T95913 CM60WQ 53361719 IC50 = 13 nM T95913 CL69DK 53377727 IC50 = 81 nM T95913 C6Q8RC 53378051 IC50 = 1584.89 nM T95913 CG3C1J 53379513 IC50 = 4.8 nM T95913 CSV9X2 54579940 IC50 = 13 nM T95913 CN51TL 54579941 IC50 = 4100 nM T95913 C7VZU2 54579942 IC50 = 2300 nM T95913 C4R9JB 54579943 IC50 = 610 nM T95913 CG26HQ 54579944 IC50 = 3700 nM T95913 CC5R3O 54580924 IC50 = 340 nM T95913 C3OIY4 54580925 IC50 = 250 nM T95913 C60TYL 54581049 IC50 = 470 nM T95913 CF2UH5 54581983 IC50 = 20 nM T95913 C23EVN 54582916 IC50 = 26 nM T95913 CT2SV7 54583916 IC50 = 480 nM T95913 CY87EC 54583917 IC50 = 30 nM T95913 C8CPI4 54584859 IC50 = 860 nM T95913 C9TZ2V 54584860 IC50 = 2300 nM T95913 CME81Q 54585830 IC50 = 190 nM T95913 CFI7E6 54754350 IC50 = 760 nM T95913 CE4TS9 56589559 IC50 = 32 nM T95913 CR24WQ 56595421 IC50 = 56 nM T95913 CJ41GT 56595686 IC50 = 52 nM T95913 C2PN4S 56599298 IC50 = 6600 nM T95913 CT64SR 56599306 IC50 = 23 nM T95913 CFUT05 56648675 IC50 = 17 nM T95913 C1GAB6 56648677 IC50 = 37 nM T95913 CWDF40 56648757 IC50 = 20 nM T95913 CE35CB 56648758 IC50 = 10 nM T95913 CJO39U 56648759 IC50 = 25 nM T95913 CNKC90 56654649 IC50 > 9100 nM T95913 C83QGP 56660108 IC50 = 9.5 nM T95913 CYM1D0 56660109 IC50 = 6 nM T95913 CHA35L 56663573 IC50 = 4 nM T95913 CF7PY5 56667023 IC50 = 7 nM T95913 CC1DJ8 56670464 IC50 = 20.5 nM T95913 CZH95G 56673952 IC50 = 8 nM T95913 CHR8K0 56677282 IC50 = 10.5 nM T95913 C79AMB 56677283 IC50 = 13.5 nM T95913 CG17TZ 56683916 IC50 = 9.5 nM T95913 C7B2OH 56683917 IC50 = 6.5 nM T95913 C6LMP8 56683918 IC50 = 14.3 nM T95913 C94JIT 56832510 Ki = 0.55 nM T95913 C0IJP8 56927258 IC50 > 6309.57 nM T95913 CM28GU 56928390 IC50 = 280 nM T95913 C9MJG4 56929824 IC50 = 50 nM T95913 CYFB96 56932203 IC50 = 63.1 nM T95913 CJ9R2C 56932209 IC50 = 630.96 nM T95913 C8C2FG 56932238 IC50 = 125.89 nM T95913 CX6Q2K 56932240 IC50 = 10 nM T95913 CPGC81 56947516 Ki = 1 nM T95913 CO6K5Q 56955953 IC50 = 441 nM T95913 CAK91L 56955954 IC50 = 18 nM T95913 C8B6JG 56955955 IC50 = 18 nM T95913 CX4W6G 57325497 IC50 = 1750 nM T95913 CVK5A3 57328247 Ki > 500 nM T95913 CW8B4D 57330208 IC50 = 850 nM T95913 C6JMN9 57345685 IC50 = 1600 nM T95913 CZ7RE0 57345686 IC50 = 1000 nM T95913 CA53SC 57351276 Ki = 183 nM T95913 C9RB7K 57391333 Ki > 500 nM T95913 CH37SE 57391335 Ki > 500 nM T95913 C1GVK3 57391362 IC50 > 4000 nM T95913 C0PR9J 57391364 IC50 > 6300 nM T95913 C6L9HO 57391365 IC50 = 3200 nM T95913 C2QX0T 57391366 IC50 = 1600 nM T95913 CLQ9J1 57391367 IC50 = 1300 nM T95913 CQ1W0C 57393124 IC50 = 7900 nM T95913 CZ0RW2 57393125 IC50 = 1600 nM T95913 COT0L2 57394595 IC50 = 19000 nM T95913 CA93ZE 57394864 IC50 = 3200 nM T95913 C6CL4F 57395172 IC50 = 980 nM T95913 CS14ZH 57396608 Ki > 500 nM T95913 CDG2F3 57396625 IC50 = 3200 nM T95913 CD73TE 57396626 IC50 > 6300 nM T95913 CQRU75 57396627 IC50 > 6300 nM T95913 CI34XH 57396628 IC50 > 6300 nM T95913 CYM02V 57397667 IC50 = 2060 nM T95913 CQO74C 57398382 Ki > 500 nM T95913 CV2Z0C 57398383 Ki > 500 nM T95913 C3Q2ZP 57398390 IC50 > 6300 nM T95913 C56TEZ 57398391 IC50 = 5000 nM T95913 CP9Q4U 57398392 IC50 = 10000 nM T95913 C0O5KE 57398393 IC50 = 320 nM T95913 C3G9HW 57399126 IC50 > 10000 nM T95913 CYE09F 57400062 IC50 = 4000 nM T95913 CN5PY7 57400063 IC50 > 7900 nM T95913 CT0Y7E 57400064 IC50 = 2500 nM T95913 C3Q2NF 57401565 IC50 = 395000 nM T95913 CRO5Z6 57401846 Ki > 500 nM T95913 CM63CS 57401865 IC50 = 1300 nM T95913 CG6M4H 57401867 IC50 > 6300 nM T95913 CP8FY5 57401868 IC50 = 1600 nM T95913 CQ5P4X 57401869 IC50 = 2500 nM T95913 CPG6N5 57402167 IC50 = 1310 nM T95913 C8LKZ3 57402168 IC50 = 1980 nM T95913 CF68RN 57403576 IC50 = 6300 nM T95913 CL2R7T 57403577 IC50 > 6300 nM T95913 CC5N9R 57403578 IC50 > 10000 nM T95913 CZ8M5F 57403579 IC50 = 1600 nM T95913 C5NT7R 57403580 IC50 = 1300 nM T95913 CHBV63 57403581 IC50 = 400 nM T95913 CAC72X 57403582 IC50 > 6300 nM T95913 CQ5Z4S 57404801 IC50 = 39.81 nM T95913 C78YHO 57404804 IC50 = 50.12 nM T95913 CNR95F 57404840 IC50 = 1900 nM T95913 CQ4E8N 57405149 IC50 = 50.12 nM T95913 CA8BT7 57405314 IC50 = 794.33 nM T95913 CI40MW 57405315 IC50 = 501.19 nM T95913 CGN72O 57405485 IC50 = 6.31 nM T95913 C5B9XS 57406164 IC50 = 3.981 nM T95913 CEI2S9 57406702 IC50 = 3162.28 nM T95913 CED47A 57410062 IC50 > 10000 nM T95913 C1BVX6 57411134 IC50 > 10000 nM T95913 C39JSW 57411135 IC50 > 10000 nM T95913 CL8F6Q 57411137 IC50 > 10000 nM T95913 CW97FT 57411139 IC50 > 10000 nM T95913 CU0R3A 57411250 IC50 > 10000 nM T95913 C6C5TU 57411252 IC50 > 10000 nM T95913 CD0W2I 57411254 IC50 = 8135 nM T95913 CW1DA3 57411255 IC50 > 10000 nM T95913 C6U4LO 57411256 IC50 > 10000 nM T95913 CP9G7L 57411366 IC50 = 4203 nM T95913 CC5DO3 57411369 IC50 > 10000 nM T95913 C56RBS 57411372 IC50 > 10000 nM T95913 CX9O3T 57411485 IC50 > 10000 nM T95913 CQBM65 57411486 IC50 > 10000 nM T95913 CK5QX7 57411488 IC50 > 10000 nM T95913 C90LNK 57411715 IC50 > 10000 nM T95913 CPXE40 57411716 IC50 > 10000 nM T95913 CE6RY5 57411836 IC50 > 10000 nM T95913 C5JOX3 57411837 IC50 > 10000 nM T95913 C0I5JM 57419280 IC50 > 10000 nM T95913 CT6XL0 57466811 Ki = 36 nM T95913 CRB5P2 57495287 IC50 > 9100 nM T95913 C59YAC 57495353 IC50 = 2230 nM T95913 CJE19S 57523686 IC50 > 10000 nM T95913 CHIU94 57545876 IC50 = 2.512 nM T95913 C0JQ8P 57584929 Ki = 36 nM T95913 CQU8A1 57585145 Ki = 36 nM T95913 C6L4FZ 57599744 IC50 = 810 nM T95913 CV9J7D 57748162 IC50 = 320 nM T95913 CL57CP 57789333 IC50 = 870 nM T95913 CZ21KP 57900314 IC50 = 2.2 nM T95913 CO20YT 58203712 IC50 = 0.6 nM T95913 C7X0OJ 58203779 IC50 = 8.4 nM T95913 CW1M9X 58203976 IC50 = 36 nM T95913 COFN62 58203995 IC50 = 80 nM T95913 C16GRS 58204034 IC50 = 19.1 nM T95913 CM62NB 58204076 IC50 = 3.5 nM T95913 CGA01N 58204242 IC50 = 4.3 nM T95913 CVR9Q2 58233988 IC50 = 25.12 nM T95913 CB9AH8 58234990 IC50 = 6000 nM T95913 CJ8YI2 58234995 IC50 = 830 nM T95913 CZF3U5 58235016 IC50 = 1000 nM T95913 CM0ND7 58235018 IC50 = 930 nM T95913 C25RXY 58235020 IC50 = 1600 nM T95913 CAY94U 58235030 IC50 = 4200 nM T95913 CAJC03 58235033 IC50 = 710 nM T95913 CN7MZ8 58235039 IC50 = 2600 nM T95913 CPW84H 58235041 IC50 = 630 nM T95913 C70CRN 58235043 IC50 = 3500 nM T95913 C5SQV3 58235052 IC50 = 700 nM T95913 CEZ4T5 58235053 IC50 = 2400 nM T95913 C82LIS 58235061 IC50 = 520 nM T95913 C3SO4E 58235062 IC50 = 530 nM T95913 CZ0SD5 58235073 IC50 = 1200 nM T95913 CQP25T 58235077 IC50 = 700 nM T95913 C0LDZ2 58235079 IC50 = 13000 nM T95913 C2YG5L 58235088 IC50 = 2600 nM T95913 CTVF29 58290044 Ki = 13 nM T95913 CJ6R8Q 59251679 IC50 = 8.2 nM T95913 CWF9Z7 59251848 Ki = 13 nM T95913 CRZ5B1 59251991 IC50 = 1190 nM T95913 C6A3KL 59293676 IC50 = 690 nM T95913 CC14ZL 59293709 IC50 = 1100 nM T95913 C0R3TX 59293715 IC50 = 1400 nM T95913 C9TVC6 59293721 IC50 = 1400 nM T95913 CZ5OV1 59293740 IC50 = 410 nM T95913 CB2Z4R 59293755 IC50 = 830 nM T95913 C8AL6C 59293763 IC50 = 610 nM T95913 CT3CF1 59477024 IC50 = 100 nM T95913 CF6YB8 59477038 IC50 = 3162.28 nM T95913 CK3H9O 59477041 IC50 = 199.53 nM T95913 C7KG5E 59477042 IC50 = 1000 nM T95913 C01DZW 59477048 IC50 = 251.19 nM T95913 CPE9X3 59507470 IC50 = 142 nM T95913 C2X8TY 59548177 Ki = 80 nM T95913 C71GBC 59548184 Ki = 7 nM T95913 CGRO45 59548196 Ki = 210 nM T95913 CD39AG 59548207 Ki = 750 nM T95913 C6KP4G 59548220 Ki = 110 nM T95913 CL82RM 59548221 Ki = 7 nM T95913 CTNU85 59548226 Ki = 54 nM T95913 CLB6N4 59548232 Ki = 1100 nM T95913 C2KBG8 59548236 Ki = 9 nM T95913 CSWV07 59548243 Ki = 130 nM T95913 CN48VL 59548245 Ki = 9 nM T95913 CMT2R0 59548250 Ki = 690 nM T95913 C3I8NE 59548256 Ki = 100 nM T95913 C8W5HT 59548263 Ki = 380 nM T95913 CT8Q5B 59548274 Ki = 8 nM T95913 CBG52T 59548278 Ki = 9 nM T95913 CVF1B2 59548283 Ki = 59 nM T95913 CY31EA 59548284 Ki = 99 nM T95913 CO4GT7 59548288 Ki = 1 nM T95913 CFR7S8 59548302 Ki = 24 nM T95913 CRE8B3 59548316 Ki = 16 nM T95913 CRM20Z 59548320 Ki = 140 nM T95913 CX1KJ9 59548322 Ki = 8 nM T95913 CJE5I4 59548341 Ki = 22 nM T95913 C8O1VS 59548349 Ki = 5 nM T95913 CE9W0K 59548355 Ki = 24 nM T95913 CWC65A 59548356 Ki = 9 nM T95913 CMKP95 59548371 Ki = 9 nM T95913 CC8UV3 59548383 Ki = 12 nM T95913 C4SN3U 59548390 Ki = 21 nM T95913 CD4ET2 59548402 Ki = 58 nM T95913 CES59T 59548403 Ki = 90 nM T95913 CE8P3G 59548407 Ki = 14 nM T95913 CO4K2W 59548419 Ki = 2.2 nM T95913 CSDB78 59548424 Ki = 8 nM T95913 C81FCQ 59548431 Ki = 9 nM T95913 CLGY34 59548453 Ki = 11 nM T95913 CBT21W 59548454 Ki = 91 nM T95913 C9DIB3 59548458 Ki = 9 nM T95913 CJT68K 59548460 Ki = 40 nM T95913 C9LFT3 59548462 Ki = 7 nM T95913 CA47YQ 59548474 Ki = 12 nM T95913 CX8C2U 59548480 Ki = 3600 nM T95913 C8S0ED 59605870 IC50 = 540 nM T95913 C4Y3GL 59609976 IC50 = 441 nM T95913 C1PC0J 59634638 IC50 = 210 nM T95913 CP2UY3 59634686 IC50 = 3530 nM T95913 C1TH2N 59634692 IC50 = 1420 nM T95913 CPA0L2 59634709 IC50 = 5360 nM T95913 C7DC6R 59662371 IC50 = 2398.83 nM T95913 C5S0FG 59662506 IC50 = 5754.4 nM T95913 CBI0M6 59688563 IC50 = 398.11 nM T95913 CUYB59 60148924 IC50 = 6600 nM T95913 CM8PD7 60150509 IC50 = 160 nM T95913 C5KD3Z 60154714 Ki > 10000 nM T95913 CS0L4D 60154996 Ki > 10000 nM T95913 C1UI3P 60155086 Ki = 2600 nM T95913 CX08ON 60155087 Ki = 480 nM T95913 CX8J1I 60155265 Ki = 9 nM T95913 CAT40I 60155266 Ki = 4 nM T95913 CD56VA 60155268 Ki = 21 nM T95913 CCQB56 60155375 IC50 = 10 nM T95913 CH5X2S 60155376 IC50 = 18 nM T95913 C74FEN 60155377 IC50 = 326 nM T95913 CZ6G4B 60155378 IC50 = 39 nM T95913 C10AHQ 60155379 IC50 = 17 nM T95913 C5FI4P 60155451 Ki = 18 nM T95913 CX9G4U 60155452 Ki = 8 nM T95913 C9Q7DE 60155469 IC50 = 26 nM T95913 CH8UY5 60155470 IC50 = 65 nM T95913 C3EDY4 60155471 IC50 = 507 nM T95913 CE0ZX1 60155472 IC50 = 152 nM T95913 CG90MC 60155473 IC50 = 53 nM T95913 C82PVI 60155474 IC50 = 167 nM T95913 CX49FT 60155475 IC50 = 161 nM T95913 CR7EG9 60155538 Ki = 46 nM T95913 CU6YB9 60155539 Ki = 30 nM T95913 CW6N1S 60155552 IC50 = 11 nM T95913 CIB08V 60155553 IC50 = 48 nM T95913 CZE28G 60155554 IC50 = 43 nM T95913 CZD2W7 60155555 IC50 = 31 nM T95913 CO6IU3 60155556 IC50 = 49 nM T95913 C6HN5O 60155557 IC50 = 18 nM T95913 CMQ9G1 60155638 IC50 = 507 nM T95913 CG56KT 60155639 IC50 = 26 nM T95913 CBJ65P 60155640 IC50 = 42 nM T95913 C8OJK0 60155641 IC50 = 5 nM T95913 CT9XJ6 60155642 IC50 = 21 nM T95913 C5BYQ3 60155643 IC50 = 8 nM T95913 C57RBF 60155722 IC50 = 587 nM T95913 CU7J6L 60155723 IC50 = 102 nM T95913 CSZA16 60155724 IC50 = 34 nM T95913 C21DWT 60155725 IC50 = 497 nM T95913 C12CQU 60155726 IC50 = 60 nM T95913 CA5TM3 60155805 IC50 = 20 nM T95913 C60RIO 60155806 IC50 = 6 nM T95913 CIRO73 66493714 IC50 = 167 nM T95913 C71LPV 66493729 IC50 = 302 nM T95913 C54NOW 66552297 IC50 > 100000 nM T95913 CX4HW1 66552298 IC50 > 50118.72 nM T95913 CEJ54A 66552343 IC50 = 501.19 nM T95913 CUQ5Y2 66552345 IC50 > 3981.07 nM T95913 C5F8ZE 66552346 IC50 > 100000 nM T95913 CHQC56 66552347 IC50 = 3162.28 nM T95913 CS6BQ0 66552348 IC50 > 12589.25 nM T95913 CGT2V9 66552407 IC50 = 3981.07 nM T95913 CIJ3C5 66552408 IC50 = 39.81 nM T95913 C6ZFI1 66552410 IC50 > 31622.78 nM T95913 C8S7CM 66552411 IC50 = 316.23 nM T95913 C9A7IK 66552412 IC50 > 39810.72 nM T95913 CRC24S 66552467 IC50 > 100000 nM T95913 CHU5V3 66552468 IC50 > 100000 nM T95913 C46POH 66552523 IC50 = 1995.26 nM T95913 C68LXT 66552524 IC50 = 25118.86 nM T95913 C91JZL 66553214 IC50 = 8280 nM T95913 CUC7B3 66557964 IC50 = 190 nM T95913 C9X2TB 66558056 IC50 = 340 nM T95913 CWZ54O 66600540 Ki = 20 nM T95913 C6Q0KU 66612050 Ki = 34 nM T95913 C1R3SI 66653673 IC50 = 3290 nM T95913 CF8BZ7 66677439 IC50 = 1060 nM T95913 C8L9DK 66743362 Ki = 14 nM T95913 C1IKT2 66743443 Ki = 11 nM T95913 CN0RE8 66779813 IC50 = 1000 nM T95913 C3IP5D 66779815 IC50 = 1000 nM T95913 CH86MR 66779905 IC50 = 1600 nM T95913 CX2N6E 66779920 IC50 > 790 nM T95913 C9O4TC 66779989 IC50 = 400 nM T95913 CF2UM8 66780001 IC50 = 4000 nM T95913 CHU0C5 66780007 IC50 = 500 nM T95913 CGL4V1 66780016 IC50 = 2000 nM T95913 C5F6OA 66780027 IC50 = 6300 nM T95913 C8DN7A 66780034 IC50 = 4000 nM T95913 C4AM6R 66780100 IC50 = 1300 nM T95913 CZ5P2N 66780118 IC50 = 160 nM T95913 CREA54 66780266 IC50 = 1300 nM T95913 CRCA72 66780292 IC50 = 2500 nM T95913 CW2SM6 66780337 IC50 = 250 nM T95913 CU54DY 66780379 IC50 = 2500 nM T95913 CQ70YA 66780434 IC50 > 7900 nM T95913 C8F9UY 66780515 IC50 = 250 nM T95913 CFH6C2 66780644 IC50 = 2500 nM T95913 CTZB46 66780835 IC50 = 7900 nM T95913 CEP5A2 66780844 IC50 > 6300 nM T95913 C51ARE 66788835 Ki = 5.3 nM T95913 C3PL1S 66800530 IC50 = 63.1 nM T95913 CJN4M2 66806967 IC50 = 630.96 nM T95913 CW12XO 66882257 IC50 > 10000 nM T95913 C6IO1S 66883557 IC50 > 10000 nM T95913 C1HSE0 67035086 IC50 = 980 nM T95913 C38RGB 67035556 IC50 > 9100 nM T95913 C5E4AJ 67050504 IC50 = 11 nM T95913 CMWO25 67061712 IC50 = 1.4 nM T95913 C0OX5N 67103709 IC50 = 1500 nM T95913 C9J2EO 67103712 IC50 = 210 nM T95913 CM4W1Y 67103722 IC50 = 2500 nM T95913 C5TYQ3 67103909 IC50 = 140 nM T95913 CVJ49E 67103974 IC50 = 1200 nM T95913 C3VFY7 67104025 IC50 = 3500 nM T95913 CC07KA 67104052 IC50 = 2900 nM T95913 C4Z0HT 67159178 IC50 <= 10000 nM T95913 C7EZW6 67192973 IC50 = 1600 nM T95913 CQHF85 67284779 IC50 = 2010 nM T95913 CT6BX3 67285457 Ki = 16000 nM T95913 C9LI0M 67294297 Ki = 49.1 nM T95913 C5BZ2V 67981475 IC50 = 1000 nM T95913 CK86XZ 67982080 IC50 = 316.23 nM T95913 CS0TY5 67982485 IC50 = 398.11 nM T95913 C9A2RD 67982543 IC50 = 3981.07 nM T95913 C7A0GH 67982639 IC50 = 1584.89 nM T95913 CW79LA 67982712 IC50 = 1258.93 nM T95913 CEG3F8 67983123 IC50 = 3000 nM T95913 C25AHY 67984037 IC50 = 8500 nM T95913 C7N4ZS 68034365 IC50 = 2400 nM T95913 CG53JO 68044823 Ki = 11 nM T95913 CGA82Q 68044837 Ki = 35 nM T95913 C4RLP9 68044907 Ki = 9 nM T95913 C6U8RP 68045063 Ki = 8 nM T95913 C0LQN1 68045070 Ki = 60 nM T95913 C7DL6V 68045162 Ki = 28 nM T95913 CA4JF3 68045179 Ki = 7 nM T95913 C57DTK 68045182 Ki = 4 nM T95913 CUQ2W1 68095924 IC50 = 158.49 nM T95913 CUR8N0 68096082 IC50 = 501.19 nM T95913 C8I7GC 68293638 IC50 > 10000 nM T95913 C45TIJ 69489467 Ki = 59.8 nM T95913 C8MTV6 70674592 IC50 = 280 nM T95913 CXB45Q 70674939 IC50 = 108 nM T95913 CAR46Z 70675172 IC50 = 72 nM T95913 CN09DI 70675846 IC50 = 97400 nM T95913 C6BQE1 70681248 IC50 = 1600 nM T95913 CPE36T 70681262 IC50 = 200 nM T95913 CPX41V 70682086 IC50 = 6.31 nM T95913 CZ5TI9 70682135 IC50 = 5120 nM T95913 CQW54O 70682591 Ki = 230 nM T95913 CPV59G 70682592 Ki = 1140 nM T95913 CB3ZN5 70683337 IC50 = 2500 nM T95913 C1I5PH 70683338 IC50 = 250 nM T95913 CSM0A6 70684204 IC50 = 2.512 nM T95913 CXD08N 70684690 Ki = 61 nM T95913 CG95EC 70684794 Ki = 84 nM T95913 C8O2QH 70685440 IC50 = 500 nM T95913 CZG9M1 70685441 IC50 = 2000 nM T95913 CH7KO0 70685442 IC50 = 1300 nM T95913 C6G4WB 70686339 IC50 = 251.19 nM T95913 CON8X4 70686340 IC50 = 63.1 nM T95913 C1ASW4 70686341 IC50 = 25.12 nM T95913 C0PWL5 70686455 IC50 = 125.89 nM T95913 CN4CR2 70686584 IC50 = 4100 nM T95913 C85FWA 70686829 Ki = 110 nM T95913 CQS8G7 70686830 Ki = 530 nM T95913 C8QSD2 70688455 IC50 = 7.943 nM T95913 CFCJ02 70688558 IC50 = 15.85 nM T95913 CSX6I7 70688908 Ki = 110 nM T95913 C1U5FC 70689024 Ki = 124 nM T95913 C5YN6U 70689166 IC50 = 5000 nM T95913 C6L4WY 70689639 IC50 = 790 nM T95913 CGT1X2 70690496 IC50 = 25.12 nM T95913 CTY78N 70690549 IC50 = 5740 nM T95913 CW3U5J 70690994 Ki = 260 nM T95913 CC6I1Q 70691259 IC50 = 3200 nM T95913 CD3JL4 70691776 IC50 = 500 nM T95913 CDK52M 70692650 IC50 = 15.85 nM T95913 CGQJ68 70692914 IC50 = 7.943 nM T95913 C7G5UV 70692915 IC50 = 7.943 nM T95913 C3TM1F 70693128 Ki = 57 nM T95913 C2VAU8 70693129 Ki = 32 nM T95913 CU3WF2 70693248 Ki = 26.7 nM T95913 C65FHO 70694723 Ki = 62.9 nM T95913 CPFO83 70694805 IC50 = 12.59 nM T95913 CRNY76 70695188 Ki = 62 nM T95913 C3N5YJ 70695189 Ki = 5810 nM T95913 C75YGN 70695469 IC50 > 3200 nM T95913 C61CFG 70696737 IC50 = 31.62 nM T95913 C7KL5X 70696852 IC50 = 125.89 nM T95913 CRH8E2 71270723 IC50 = 501.19 nM T95913 CWR58A 71270783 IC50 > 1479.11 nM T95913 CF9LU4 71270807 IC50 = 501.19 nM T95913 C7FDL2 71270817 IC50 = 398.11 nM T95913 CNR1G9 71270824 IC50 = 2511.89 nM T95913 C38LBA 71270831 IC50 = 316.23 nM T95913 CTL6R5 71270836 IC50 = 398.11 nM T95913 CM4LX7 71270848 IC50 > 6309.57 nM T95913 C2GWX6 71270906 IC50 = 1995.26 nM T95913 CX0DL3 71270910 IC50 > 3981.07 nM T95913 C0COW6 71270913 IC50 > 6309.57 nM T95913 CB0S8G 71270927 IC50 = 251.19 nM T95913 C24IOW 71270948 IC50 > 5011.87 nM T95913 C5BJ2Y 71270957 IC50 > 3162.28 nM T95913 C03NFY 71271625 IC50 > 5011.87 nM T95913 CL47JU 71271739 IC50 > 7943.28 nM T95913 CS5JG6 71271910 IC50 > 6309.57 nM T95913 C4PSK8 71271965 IC50 = 316.23 nM T95913 CB4N1M 71272066 IC50 > 5011.87 nM T95913 CD8E1Y 71272453 IC50 = 630.96 nM T95913 C8EW9V 71272757 IC50 = 3162.28 nM T95913 C0LO8I 71272765 IC50 = 398.11 nM T95913 C1MVL0 71273460 Ki = 40.6 nM T95913 CK58RV 71449587 IC50 = 91 nM T95913 C0ROQ6 71450451 IC50 = 22 nM T95913 CTL30H 71450452 IC50 = 12 nM T95913 CNX18D 71450453 IC50 = 24 nM T95913 C7HT4F 71450454 IC50 = 46 nM T95913 CNHJ63 71451228 IC50 = 777 nM T95913 CD8Y3S 71451617 Ki = 2350 nM T95913 C9SC2V 71452282 IC50 = 16 nM T95913 CY62VF 71452283 IC50 = 181 nM T95913 CQ7C5R 71452284 IC50 = 14 nM T95913 C6VF7J 71453206 IC50 = 63 nM T95913 CR84JX 71453419 Ki = 4 nM T95913 CZ61FJ 71454160 IC50 = 25.12 nM T95913 CZ8Q5P 71454238 Ki = 2.4 nM T95913 CF74SL 71454944 IC50 = 93 nM T95913 CO82IY 71455167 Ki = 21 nM T95913 CA7L1Y 71455168 Ki = 31 nM T95913 CSW47K 71455817 IC50 = 117 nM T95913 CT32GB 71455818 IC50 = 10 nM T95913 CE1IX7 71456728 IC50 = 59 nM T95913 CLUR84 71457607 IC50 = 12 nM T95913 C4ACV9 71457608 IC50 = 95 nM T95913 CM1ND2 71458573 IC50 = 82 nM T95913 C3S0NP 71458574 IC50 = 72 nM T95913 CY6WI2 71458575 IC50 = 60 nM T95913 C13KJV 71459500 IC50 = 250 nM T95913 CO8U5R 71459501 IC50 = 223 nM T95913 CL30DJ 71459502 IC50 = 346 nM T95913 C1Y8WD 71459503 IC50 = 12 nM T95913 CT7K3A 71460422 IC50 = 54 nM T95913 CW9YM2 71461240 IC50 = 3 nM T95913 CA2V9S 71461241 IC50 = 161 nM T95913 C65RJY 71461242 IC50 = 25 nM T95913 C2HOB7 71461243 IC50 = 3 nM T95913 CO26VM 71462973 IC50 = 24 nM T95913 CU3EO6 71520393 IC50 > 10000 nM T95913 CYC6S1 71520394 IC50 > 10000 nM T95913 C1KMX0 71520395 IC50 > 10000 nM T95913 CYK7N8 71520396 IC50 > 10000 nM T95913 CTC0O8 71520397 IC50 > 10000 nM T95913 C0UZ3D 71526877 IC50 = 2000 nM T95913 CP05SQ 71526878 IC50 = 100000 nM T95913 CZK6X9 71526879 IC50 > 10000 nM T95913 C8QRE4 71526880 IC50 > 10000 nM T95913 CT3QI8 71526881 IC50 > 10000 nM T95913 CO4MY1 71527005 IC50 > 10000 nM T95913 CJC64F 71527006 IC50 > 10000 nM T95913 C96WZG 71527007 IC50 = 3900 nM T95913 CUC7I1 71527008 IC50 = 8000 nM T95913 C09WKC 71527009 IC50 > 10000 nM T95913 CSPO76 71527716 IC50 > 5011.87 nM T95913 CIN7O1 71527842 IC50 > 6309.57 nM T95913 CO6CI7 71528725 IC50 = 9900 nM T95913 C5U2ZC 71528726 IC50 = 380 nM T95913 CTKO36 71528727 IC50 = 3600 nM T95913 C2KF3X 71533728 IC50 = 1046 nM T95913 CI7Q4K 71548718 IC50 = 2700 nM T95913 CED62L 71548719 IC50 = 9200 nM T95913 C4B0KN 71549093 IC50 = 20000 nM T95913 C6PRV1 71655831 IC50 = 12 nM T95913 CU48RN 71657825 IC50 = 154 nM T95913 CWG8M3 71682651 IC50 = 210 nM T95913 C6UGW3 71682652 IC50 = 4600 nM T95913 C7BX4K 71682653 IC50 = 930 nM T95913 CQX8N3 71682654 IC50 > 10000 nM T95913 CS32HB 71716798 IC50 > 6309.57 nM T95913 C07GCV 71716799 IC50 = 5011.87 nM T95913 CFW01E 71718034 IC50 = 2530 nM T95913 CXJC41 72188489 IC50 = 1000 nM T95913 C29KOU 72709209 IC50 > 10000 nM T95913 CT73IW 72709284 IC50 = 2500 nM T95913 CIL6S8 72737375 IC50 = 28 nM T95913 CTYJ25 72737376 IC50 = 158 nM T95913 CPL27S 72737377 IC50 = 52 nM T95913 C5RQB7 72737378 IC50 = 68 nM T95913 C8H7VT 72737379 IC50 = 121 nM T95913 CV2G1F 72737380 IC50 = 62 nM T95913 CHX84Q 72737381 IC50 = 7.2 nM T95913 CI5OT1 72737382 IC50 = 203 nM T95913 CSN5U8 72737551 IC50 = 17 nM T95913 CHC5J2 72737552 IC50 = 29 nM T95913 CB5PM9 72737553 IC50 = 68 nM T95913 CIF36E 72737554 IC50 = 57 nM T95913 C87HDL 72737555 IC50 = 100 nM T95913 CVU2J9 72949025 IC50 = 42 nM T95913 CC6KY3 72949203 IC50 = 16 nM T95913 CYGV85 73051332 IC50 = 5 nM T95913 CV4BH5 73051810 IC50 = 34 nM T95913 CE2IG4 73051811 IC50 = 271 nM T95913 CKUF15 73051812 IC50 = 4 nM T95913 CRF25X 73051813 IC50 = 12 nM T95913 C56JVH 73051977 IC50 = 67 nM T95913 C7N0AF 73052137 IC50 = 11 nM T95913 CNTD65 73052455 IC50 = 6 nM T95913 CZY9U8 73441896 IC50 = 31622.78 nM T95913 CL0XZ1 73659199 Ki = 2 nM T95913 CK7XM5 73659200 Ki = 1 nM T95913 C8EI1X 73673707 IC50 = 1.5 nM T95913 C0W1TK 73774799 IC50 = 120 nM T95913 C4W3IL 73774944 IC50 = 420 nM T95913 CH75QS 73774946 IC50 = 11 nM T95913 C5NKS4 73774948 IC50 = 40 nM T95913 C23MSN 73775105 IC50 = 160 nM T95913 CQG43I 73775546 IC50 = 3.3 nM T95913 CBXV38 73775549 IC50 = 3.1 nM T95913 C6O4PV 73775675 IC50 = 15 nM T95913 CQI4G9 73775798 IC50 = 81 nM T95913 CG0VK1 73775800 IC50 = 17 nM T95913 C7N0ME 73775931 IC50 = 3.6 nM T95913 CA5DJ3 73775934 IC50 = 13 nM T95913 CD6M4Q 73776065 IC50 = 10 nM T95913 C6X3LA 73776070 IC50 = 0.3 nM T95913 C5PKH6 73776209 IC50 = 430 nM T95913 C4WLT1 73776507 IC50 = 12 nM T95913 CPH39S 73776508 IC50 = 45 nM T95913 CT6ZB1 73776511 IC50 = 64 nM T95913 CI9K0J 73776652 IC50 = 0.7 nM T95913 CMHK83 73776786 IC50 = 0.6 nM T95913 CMT13V 73776787 IC50 = 6.8 nM T95913 CBYN18 73977439 IC50 = 1995 nM T95913 C9V1YR 73977449 IC50 = 251 nM T95913 CXA90D 73977451 IC50 = 316 nM T95913 CEZ7L2 73977461 IC50 = 126 nM T95913 CD0T9V 74539799 IC50 = 0.74 nM T95913 C16KOS 74539862 IC50 = 1.1 nM T95913 CN2MI8 76310247 IC50 > 50000 nM T95913 CKO41J 76310248 IC50 = 741 nM T95913 CEN9Q5 76310249 IC50 > 50000 nM T95913 CJCF67 76310250 IC50 = 26 nM T95913 CBF70W 76310805 IC50 = 316.23 nM T95913 CA2VR6 76311340 IC50 = 194.98 nM T95913 CMR07I 76313939 IC50 > 50000 nM T95913 C5P2CJ 76313940 IC50 = 30700 nM T95913 CAV5Q9 76313941 IC50 = 22000 nM T95913 CO13XZ 76314937 IC50 = 386 nM T95913 C7W2HI 76314938 IC50 = 341.98 nM T95913 C6H9EL 76314939 IC50 = 230.99 nM T95913 C0J6PL 76317466 IC50 > 50000 nM T95913 CVW35P 76317467 IC50 > 50000 nM T95913 CZ1T3C 76317468 IC50 > 50000 nM T95913 C4MKN3 76317469 IC50 = 62 nM T95913 C3JA4F 76317470 IC50 = 353 nM T95913 C4XJ5Y 76317471 IC50 = 153 nM T95913 CS6ME5 76318566 IC50 = 235 nM T95913 CG4I2R 76318567 IC50 = 217 nM T95913 C8E4GI 76321204 IC50 = 183 nM T95913 CF4OI8 76321205 IC50 = 12300 nM T95913 C1YFK9 76322218 IC50 = 267.98 nM T95913 CL0T7B 76322219 IC50 <= 65 nM T95913 CDG8V4 76324821 IC50 = 87 nM T95913 CJW39V 76324822 IC50 > 50000 nM T95913 C2BFA1 76324823 IC50 = 4700 nM T95913 CM4N8A 76325342 IC50 = 6309.57 nM T95913 C92ZAB 76325343 IC50 = 25118.86 nM T95913 C1HFI9 76325446 IC50 = 3259 nM T95913 C4GZ1Q 76325833 IC50 = 357.03 nM T95913 CQ31CA 76325834 IC50 = 312.97 nM T95913 C4A8XZ 76328376 IC50 = 3400 nM T95913 C39CLE 76329428 IC50 = 247 nM T95913 CYR0G6 76332050 IC50 = 6300 nM T95913 C4MID5 76332051 IC50 = 7880 nM T95913 C70WJE 76332052 IC50 = 79 nM T95913 CQ8YC1 76332568 IC50 = 7.943 nM T95913 CE6BI0 76332666 IC50 = 4350 nM T95913 C16SRX 76333068 IC50 = 143 nM T95913 CW81MC 76333069 IC50 = 264.97 nM T95913 C26CKL 76333070 IC50 = 153.99 nM T95913 C47NLT 76333071 IC50 = 250 nM T95913 CN38BK 76335378 IC50 = 81 nM T95913 C69ATM 76335666 IC50 > 50000 nM T95913 C0SI4C 76335667 IC50 > 50000 nM T95913 C31NEK 76335668 IC50 = 574 nM T95913 CL6BV5 76335669 IC50 > 50000 nM T95913 C73KJD 76335670 IC50 = 227 nM T95913 CY3LO5 76336173 IC50 = 1258.93 nM T95913 CJ3V6Y 76336695 IC50 = 274 nM T95913 CD03GB 76336696 IC50 = 277.97 nM T95913 C2JTH8 77107528 IC50 = 112 nM T95913 C42HDP 77107927 IC50 = 42 nM T95913 C04SRC 77147259 IC50 = 1774 nM T95913 C9I7TY 78319187 IC50 = 1584.89 nM T95913 C24LQH 78320362 IC50 = 35 nM T95913 C9T8KF 78320671 IC50 = 70 nM T95913 CI2YN8 78320672 IC50 = 24 nM T95913 CI6K4J 78320673 IC50 = 305 nM T95913 COFJ16 78320996 IC50 = 5200 nM T95913 CMU5P2 78321310 IC50 = 150 nM T95913 CE13AJ 78321314 IC50 = 200 nM T95913 CSP2H4 78321635 IC50 = 280 nM T95913 CWA0B1 78322567 IC50 = 140 nM T95913 CH6P9D 78322877 IC50 > 10000 nM T95913 C4IW9V 78323193 IC50 = 230 nM T95913 CD1JC8 78324443 IC50 = 129 nM T95913 C04IKP 86268622 IC50 = 28 nM T95913 C5P3RO 86647783 IC50 = 1200 nM T95913 CDXM47 86677874 IC50 > 10000 nM T95913 CP3W1B 86695297 IC50 > 20000 nM T95913 CA17UE 86732669 IC50 = 4630 nM T95913 C2PCS7 87061302 IC50 = 181 nM T95913 CNVS32 87343636 Ki = 16.7 nM T95913 CV6PI8 87562294 IC50 = 125.89 nM T95913 CZ2AU4 87570781 IC50 = 375 nM T95913 C3HD5O 88570842 Ki = 9 nM T95913 CLEX32 89034287 Ki = 4 nM T95913 C1AKZ4 89034365 Ki = 6 nM T95913 CEQ80V 89034380 Ki = 5 nM T95913 C1HB3F 89051931 IC50 = 330 nM T95913 C61SCX 89493851 IC50 = 5 nM T95913 C1LU3X 89493904 IC50 = 31 nM T95913 CTE1L0 89517065 IC50 = 9300 nM T95913 C56KSC 89517226 IC50 > 10000 nM T95913 C6M0QF 89841854 IC50 = 400 nM T95913 C61GIO 89841941 IC50 = 40 nM T95913 C6FI0A 89842032 IC50 = 110 nM T95913 COL45N 89842055 IC50 = 60 nM T95913 C7FNP8 89842123 IC50 = 25 nM T95913 CF50MO 89842136 IC50 = 1100 nM T95913 C6CKP2 89842150 IC50 = 50 nM T95913 CVZH15 89842186 IC50 = 240 nM T95913 C2LQ9V 89842220 IC50 = 150 nM T95913 C83SXM 89842240 IC50 = 1100 nM T95913 CQ1U2Y 89842245 IC50 = 1000 nM T95913 CQO85K 89842249 IC50 > 7000 nM T95913 CX70NQ 89842250 IC50 = 14 nM T95913 CN5Y9A 90064110 IC50 = 27 nM T95913 C7FP2M 90064111 IC50 = 4 nM T95913 CN51BK 90064299 IC50 = 2 nM T95913 CUZ13D 90102336 IC50 = 0.7 nM T95913 CQO9J0 90103194 IC50 = 1.7 nM T95913 C28WQY 90431726 IC50 = 20 nM T95913 C08UWK 90665816 IC50 = 100000 nM T95913 CMWB58 91757958 IC50 <= 10000 nM T95913 C3Y0DS 91801158 IC50 = 2.6 nM T95913 CAS7W6 91864650 IC50 = 8440 nM T95913 CA3ZC1 92172785 IC50 = 575000 nM T95913 C4JMV1 118003503 IC50 = 330 nM T95913 C6YRW7 118003617 IC50 = 110 nM T95913 C8QHY9 118003714 IC50 = 75 nM T95913 CLDA15 118003719 IC50 = 360 nM T95913 C5LW9G 118004010 IC50 = 100 nM T95913 CK0W1T 118004012 IC50 = 170 nM T95913 C0BIP8 118004016 IC50 = 350 nM T95913 CB4PM3 118004022 IC50 = 110 nM T95913 CNCK58 118004064 IC50 = 280 nM T95913 C14WCU 118131317 IC50 > 1000 nM T95913 C67VQE 118341819 IC50 = 850 nM T95913 CC9P5H 118341835 IC50 = 750 nM T95913 CUMA23 118341844 IC50 = 1840 nM T95913 C3IP9X 118341852 IC50 = 190 nM T95913 C6TI0Z 118341865 IC50 = 520 nM T95913 C4U7NC 118341870 IC50 = 360 nM T95913 CVL03K 118341884 IC50 = 1370 nM T95913 CPZN96 118341923 IC50 = 150 nM T95913 C9E3DU 118341927 IC50 = 6950 nM T95913 CVN87P 118433737 IC50 = 36 nM T95913 C8W1RN 118445922 IC50 = 7 nM T95913 CGYA58 118445928 IC50 = 182 nM T95913 CL29BI 118445929 IC50 = 52 nM T95913 CI24WZ 118445978 IC50 = 3 nM T95913 CA20CO 118445983 IC50 = 13 nM T95913 CQF1V4 118446049 IC50 = 4 nM T95913 C90OAT 118446064 IC50 = 43 nM T95913 CJQ92T 118572891 IC50 < 10 nM T95913 CVY45K 118575373 IC50 > 10000 nM T95913 CS20UM 118575423 IC50 > 10000 nM T95913 CCPV26 118575517 IC50 = 632 nM T95913 C0L9JQ 118575526 IC50 = 1300 nM T95913 CH6AB7 118575540 IC50 > 10000 nM T95913 C97QIN 118575555 IC50 = 990 nM T95913 CEDC48 118575654 IC50 = 3466 nM T95913 COYJ84 118575663 IC50 > 10000 nM T95913 CS1Z8W 118575682 IC50 = 4407 nM T95913 CC0S4G 118575689 IC50 = 199 nM T95913 C6X8HG 118575694 IC50 > 10000 nM T95913 CUJ30I 118575784 IC50 = 1247 nM T95913 CAT54V 118575791 IC50 = 1277 nM T95913 C1K6HU 118575835 IC50 = 4262 nM T95913 C2OQ4U 118575893 IC50 > 10000 nM T95913 C6HEA7 118575940 IC50 = 990 nM T95913 CIU7J3 118575971 IC50 = 267 nM T95913 CAD39P 118575986 IC50 = 4150 nM T95913 CCYI54 118576050 IC50 = 1131 nM T95913 CW9T6F 118576060 IC50 = 7836 nM T95913 C7Y4AT 118576103 IC50 > 10000 nM T95913 C47WMX 118576166 IC50 = 7989 nM T95913 C1UT8B 118576192 IC50 > 10000 nM T95913 C0F7JV 118576207 IC50 = 2311 nM T95913 CU61WD 118576212 IC50 > 10000 nM T95913 CE3V8W 118576268 IC50 = 54 nM T95913 CO0YC8 118616775 IC50 = 1 nM T95913 CS5C8W 118684133 IC50 = 4.3 nM T95913 CRX24W 118709077 IC50 = 6000 nM T95913 CV2EJ7 118709081 IC50 = 6900 nM T95913 CZ41AQ 118709092 IC50 = 83000 nM T95913 CR6ML1 118709578 IC50 = 670 nM T95913 C0OH7I 118709579 IC50 = 13500 nM T95913 C73YIO 118709582 IC50 = 3000 nM T95913 CGWX02 118709583 IC50 = 510 nM T95913 CY2QG0 118711873 IC50 = 10890 nM T95913 CH4XY2 118711874 IC50 = 10710 nM T95913 C94GZM 118712046 IC50 = 3600 nM T95913 CPXQ86 118721834 Ki = 44 nM T95913 CH9D8G 118721835 Ki = 19 nM T95913 CYHG95 118721836 Ki = 21 nM T95913 CP6SR7 118721837 Ki = 9 nM T95913 CW4N7Q 118721838 Ki = 7 nM T95913 CZG78A 118721839 Ki = 190 nM T95913 C2BQS3 118721840 Ki = 6 nM T95913 C2T9RN 118721841 Ki = 1 nM T95913 C6GJ0Q 118721842 Ki = 7 nM T95913 C9RPN4 118721843 Ki = 2 nM T95913 CYNZ53 118721844 Ki = 22 nM T95913 C5R1VP 118721845 Ki = 19 nM T95913 CB53EU 118728320 IC50 = 34624 nM T95913 C6KJL1 118728321 IC50 = 21668 nM T95913 CKJ3S6 118728322 IC50 = 27916 nM T95913 CT0L3Y 118728325 IC50 = 24342 nM T95913 CHS2E4 118728326 IC50 = 11812 nM T95913 CRUP47 118728328 IC50 = 44117 nM T95913 CQR41G 118728330 IC50 = 19479 nM T95913 CN4Q9R 118728332 IC50 = 9443 nM T95913 CDI10F 118728336 IC50 = 41626 nM T95913 CHT6K9 118728811 Ki = 2900 nM T95913 CUA3Y2 118728812 Ki > 4000 nM T95913 CDQ78G 118728813 Ki = 400 nM T95913 CZ6XL7 118728814 Ki = 630 nM T95913 CMO67K 118728815 Ki = 750 nM T95913 CR2M0Q 118728816 Ki = 1500 nM T95913 C62SCL 118728817 Ki = 690 nM T95913 CSB30C 118728819 Ki = 1100 nM T95913 CV7XU8 118728820 Ki = 710 nM T95913 C3J1EX 118728821 Ki > 4000 nM T95913 CIWB78 118728822 Ki > 4000 nM T95913 CP18SE 118728823 Ki = 780 nM T95913 CM42CA 118728824 Ki = 1400 nM T95913 C9Q7CL 118728825 Ki = 2800 nM T95913 CCR3S0 118728826 Ki = 1200 nM T95913 CB1WC5 118729946 IC50 = 380 nM T95913 CQ4G9M 118729947 IC50 = 1600 nM T95913 C43IPJ 118729948 IC50 = 250 nM T95913 C3I9CQ 118729949 IC50 = 510 nM T95913 CZQ17M 118729950 IC50 = 200 nM T95913 C3G1ZP 118729951 IC50 = 4950 nM T95913 CY60FC 118730033 IC50 = 17087 nM T95913 CN3B4U 118730711 IC50 = 320 nM T95913 C0IL3N 118730712 IC50 = 1400 nM T95913 C3CH1A 118730713 IC50 = 350 nM T95913 CHX5L9 118730714 IC50 = 250 nM T95913 CNJ32C 118730715 IC50 = 3200 nM T95913 C1MKB3 118730716 IC50 = 1400 nM T95913 C81RJA 118730717 IC50 = 13000 nM T95913 CFZ16R 118737301 IC50 <= 10000 nM T95913 C27CPQ 118737302 IC50 <= 10000 nM T95913 C59VXA 118737303 IC50 <= 10000 nM T95913 CGO1N4 118737304 IC50 <= 10000 nM T95913 CS85FM 118737305 IC50 <= 10000 nM T95913 C8UCO1 118737306 IC50 <= 10000 nM T95913 CR0BZ2 118737307 IC50 <= 10000 nM T95913 C3N4DJ 118737308 IC50 <= 10000 nM T95913 CGY5B1 118737309 IC50 <= 10000 nM T95913 CV85EL 118981804 IC50 = 38 nM T95913 C91PVZ 121428416 IC50 = 204 nM T95913 CA2DM0 121428489 IC50 = 164 nM T95913 CQLX36 121428567 IC50 = 288 nM T95913 CFN12W 121445751 IC50 = 28 nM T95913 C04NDW 121445810 IC50 = 41 nM T95913 C81IFQ 122163152 IC50 = 1340 nM T95913 C2VGD5 122178120 IC50 = 21.1 nM T95913 C24XUZ 122178124 IC50 = 10.2 nM T95913 CN5AB3 122179486 IC50 = 4.4 nM T95913 CLEK13 122179487 IC50 = 10 nM T95913 C0OW8H 122179490 IC50 = 52 nM T95913 C0VD5F 122179491 IC50 = 2 nM T95913 CQ87FB 122179492 IC50 = 4 nM T95913 CBJ29X 122179493 IC50 > 10000 nM T95913 CA5N1B 122179494 IC50 = 25 nM T95913 CM4AW9 122180514 Ki = 0.024 nM T95913 CM89OL 122180515 Ki = 0.016 nM T95913 CU0C1D 122180516 Ki = 0.01 nM T95913 CB6PR7 122180517 Ki = 0.034 nM T95913 CQ63DW 122180518 Ki = 0.006 nM T95913 C9N8JT 122180519 Ki = 0.003 nM T95913 C42GSX 122180520 Ki = 0.002 nM T95913 CVA3P2 122180521 Ki = 0.009 nM T95913 C0A7CQ 122180522 Ki = 0.025 nM T95913 CEFS13 122180793 IC50 = 91560 nM T95913 CFZ2E1 122180794 IC50 = 125800 nM T95913 C5YKG7 122180795 IC50 = 465500 nM T95913 C9ID7U 122180796 IC50 = 345900 nM T95913 C08XOC 122180839 IC50 = 781500 nM T95913 C2HM6P 122180840 IC50 = 967700 nM T95913 CT9Y6U 122180841 IC50 = 23640 nM T95913 C6FOM0 122180842 IC50 = 18480 nM T95913 COX90L 122180843 IC50 = 12570 nM T95913 CP40RU 122180844 IC50 = 26870 nM T95913 CC0EK9 122180845 IC50 = 15560 nM T95913 CS85CU 122181413 IC50 = 280 nM T95913 CQS67B 122181416 IC50 = 650 nM T95913 C58XRY 122184465 IC50 = 1995.26 nM T95913 C16ALM 122184466 IC50 = 1000 nM T95913 CDZY02 122184468 IC50 = 50118.72 nM T95913 CTH70U 122184469 IC50 = 12589.25 nM T95913 C9ZXR7 122184470 IC50 = 3981.07 nM T95913 CNJ9Z4 122184471 IC50 = 3981.07 nM T95913 CS41EG 122184473 IC50 = 1258.93 nM T95913 CZ36GL 122184474 IC50 = 1000 nM T95913 CU4ZT6 122184475 IC50 = 10000 nM T95913 C3H9PR 122184476 IC50 = 1258.93 nM T95913 CU40TW 122184477 IC50 = 3162.28 nM T95913 CAMD31 122184479 IC50 = 19952.62 nM T95913 C1F9RK 122184480 IC50 = 251.19 nM T95913 C7XW1K 122184481 IC50 = 12589.25 nM T95913 CRUX54 122184482 IC50 = 31622.78 nM T95913 CQ7W0P 122184526 IC50 = 3981.07 nM T95913 CA5YB2 122184529 IC50 = 2511.89 nM T95913 C64YPH 122184530 IC50 = 2511.89 nM T95913 C4AGX5 122184531 IC50 = 3162.28 nM T95913 CQL4K5 122184532 IC50 = 1584.89 nM T95913 CRKV74 122184533 IC50 = 3981.07 nM T95913 CX14YD 122184534 IC50 = 1000 nM T95913 CM6A4S 122184535 IC50 = 1258.93 nM T95913 CF86YS 122184536 IC50 = 1995.26 nM T95913 CYRH97 122184538 IC50 = 3162.28 nM T95913 CD4W0Z 122184539 IC50 = 10000 nM T95913 CH8Y3Q 122184540 IC50 = 15848.93 nM T95913 CDA85R 122184541 IC50 = 63095.73 nM T95913 CF36XJ 122184542 IC50 > 199526.23 nM T95913 CQ6O7H 122184543 IC50 = 50118.72 nM T95913 CS4MN0 122184544 IC50 = 10000 nM T95913 CKT74G 122185265 IC50 = 14 nM T95913 CJ6C1O 122185267 IC50 = 22 nM T95913 CGW35U 122387497 IC50 = 259 nM T95913 C38BML 122387499 IC50 = 265 nM T95913 CCW0M1 122387500 IC50 = 174 nM T95913 CKA90Y 122387501 IC50 = 89 nM T95913 CH4LC6 122387502 IC50 = 56 nM T95913 C8OC3E 122387504 IC50 = 169 nM T95913 C34AHY 122387505 IC50 = 185 nM T95913 CUG1T6 122387506 IC50 = 98 nM T95913 CE7K5C 122387507 IC50 = 173 nM T95913 C4HL3N 122387508 IC50 = 111 nM T95913 CA7L3S 122387509 IC50 = 112 nM T95913 CR9NF3 122542400 IC50 = 5.7 nM T95913 CZE35C 122648343 IC50 > 10000 nM T95913 C54RNT 122648367 IC50 > 10000 nM T95913 C1UVI7 122648600 IC50 = 255 nM T95913 CMX59K 122648648 IC50 = 8.1 nM T95913 CVZ64I 122648649 IC50 > 10000 nM T95913 CPTY78 124518210 IC50 = 89 nM T95913 CB7G5E 126476620 IC50 = 501.19 nM T95913 C74BNR 126480568 IC50 = 1584.89 nM T95913 C1N6YP 126480569 IC50 = 2511.89 nM T95913 CE52HC 126480570 IC50 = 630.96 nM T95913 CQ74WU 126480571 IC50 = 3981.07 nM T95913 C0AFE2 126480572 IC50 = 1000 nM T95913 C3E7JB 126480573 IC50 = 6309.57 nM T95913 CPW54V 126480574 IC50 = 1000 nM T95913 CVJ3Q5 127025094 IC50 = 285 nM T95913 C2E4LO 127025141 IC50 = 6570 nM T95913 CO94KJ 127025144 IC50 > 25000 nM T95913 CKO53P 127025146 IC50 = 21450 nM T95913 CF7H0V 127025161 IC50 = 1260 nM T95913 CE4C3J 127025163 IC50 = 12360 nM T95913 CAV24Z 127025164 IC50 = 9360 nM T95913 C98DKI 127025346 IC50 = 4 nM T95913 CDZ56M 127025449 IC50 > 25000 nM T95913 CBXJ67 127025628 IC50 = 2.7 nM T95913 CH2Q7A 127027634 IC50 = 280 nM T95913 CSV3R7 127029064 IC50 = 64 nM T95913 CQTG79 127029604 IC50 = 279 nM T95913 CZHT45 127031017 IC50 = 3700 nM T95913 CU0F4R 127031332 IC50 = 1500 nM T95913 C2IN4Q 127031333 IC50 > 50000 nM T95913 CS12RU 127031435 IC50 = 2.3 nM T95913 CGU4H3 127031891 IC50 = 21 nM T95913 CGKR53 127032915 IC50 = 502 nM T95913 C41YQI 127035981 IC50 = 939 nM T95913 C7V4WA 127036623 IC50 = 13780 nM T95913 CJ1LH4 127036935 IC50 = 3120 nM T95913 CG8DA9 127045861 IC50 = 99 nM T95913 CVF8Z9 127045862 IC50 = 5 nM T95913 CH68NT 127046076 IC50 = 77 nM T95913 CA2XD5 127046077 IC50 = 230 nM T95913 COJ68G 127046117 IC50 = 1900 nM T95913 C34REM 127046317 IC50 = 570 nM T95913 CC4ND8 127046862 IC50 = 302 nM T95913 CY2P1X 127047138 IC50 = 440 nM T95913 CZ2R0C 127047140 IC50 = 120 nM T95913 CT89GI 127047683 IC50 = 720 nM T95913 C7D0FN 127047685 IC50 = 240 nM T95913 CN94CQ 127047797 IC50 = 140 nM T95913 C3IC2Z 127052212 IC50 = 5803 nM T95913 CN9XL1 129262531 IC50 = 90 nM T95913 CW7A5X 129626595 IC50 = 3981.07 nM T95913 C18NHD 130302549 IC50 <= 10000 nM T95913 CL13RZ 130302558 IC50 <= 10000 nM T95913 CF5JZ3 130302563 IC50 <= 10000 nM T95913 CD46EL 130302605 IC50 <= 10000 nM T95913 CNI8M6 130302620 IC50 <= 10000 nM T95913 CI6WN9 130302651 IC50 <= 10000 nM T95913 C5ZP0L 130302658 IC50 <= 10000 nM T95913 CW61SG 130302663 IC50 <= 10000 nM T95913 CB27ZG 130302668 IC50 <= 10000 nM T95913 C5VYM6 130302674 IC50 <= 10000 nM T95913 C0FQR2 130302675 IC50 <= 10000 nM T95913 CB34HQ 130302676 IC50 <= 10000 nM T95913 CQR1I8 130302685 IC50 <= 10000 nM T95913 C17DZF 130302698 IC50 <= 10000 nM T95913 CBC6W7 130302701 IC50 <= 10000 nM T95913 CBT21G 130302702 IC50 <= 10000 nM T95913 CDZ45O 130302703 IC50 <= 10000 nM T95913 C2GWU8 130302709 IC50 <= 10000 nM T95913 CV3M6Y 130302710 IC50 <= 10000 nM T95913 C39UQN 130302731 IC50 <= 10000 nM T95913 CL9O8X 130302732 IC50 <= 10000 nM T95913 CL69GM 130302740 IC50 <= 10000 nM T95913 CH8YK9 130302741 IC50 <= 10000 nM T95913 CQR2W9 130302781 IC50 <= 10000 nM T95913 C9HC8A 130302803 IC50 <= 10000 nM T95913 CIK25W 130302809 IC50 <= 10000 nM T95913 CI08PF 130332501 IC50 <= 10000 nM T95913 C1H4UT 130332505 IC50 <= 10000 nM T95913 CZPI64 130332579 IC50 <= 10000 nM T95913 CDS9F3 130332582 IC50 <= 10000 nM T95913 C3G0HF 130332585 IC50 <= 10000 nM T95913 CX13UC 130332620 IC50 <= 10000 nM T95913 CED6F3 130332657 IC50 <= 10000 nM T95913 C73KWM 130338615 IC50 = 100 nM T95913 CLC06T 130406587 IC50 = 1 nM T95913 C47CAY 130421765 IC50 = 0.631 nM T95913 C84YKI 130422161 IC50 = 0.7943 nM T95913 C2MVE6 130422162 IC50 = 0.631 nM T95913 CK68CA 130453737 IC50 = 3000 nM T95913 CUO41K 130470684 IC50 = 7100 nM T95913 CDE7T3 132005217 IC50 = 49 nM T95913 CL26YS 132005219 IC50 = 310 nM T95913 CP32GB 132005220 IC50 = 15 nM T95913 CG1NC4 132005221 IC50 = 3300 nM T95913 C0UV2M 132005224 IC50 = 58 nM T95913 CUN18W 132005225 IC50 = 6.5 nM T95913 CD84OI 132005228 IC50 = 2.8 nM T95913 C9VDI0 132005229 IC50 = 110 nM T95913 CB1Z7P 132005231 IC50 = 340 nM T95913 C7ASP9 132005246 IC50 = 11 nM T95913 C8VE6T 132005248 IC50 = 560 nM T95913 C7LCW1 132005249 IC50 = 110 nM T95913 C5W9LN 132005323 IC50 = 120 nM T95913 CQ6GO2 132005326 IC50 = 330 nM T95913 C6OXE3 132134663 IC50 = 10 nM T95913 C4M8WN 132209922 IC50 = 1.3 nM T95913 CFI23B 132210082 IC50 = 21 nM T95913 C8RK4V 132218631 IC50 = 300 nM T95913 CZD9F3 132219135 IC50 > 10000 nM T95913 CH8DP7 132220479 IC50 = 41 nM T95913 C4Q5LF 132471857 IC50 = 10 nM T95913 CJE34F 132597748 IC50 = 3220 nM T95913 CCV46G 132606879 IC50 = 199.53 nM T95913 CT2PN8 132990561 IC50 = 75 nM T95913 CFG90E 134132909 IC50 = 642 nM T95913 CI49TK 134133218 IC50 = 65 nM T95913 C4YNH0 134134126 IC50 = 698 nM T95913 C0EK8P 134134680 IC50 = 828 nM T95913 C0A1UM 134138053 IC50 = 282 nM T95913 CQ2S4X 134138703 IC50 > 9100 nM T95913 CL3Q6G 134140420 IC50 = 1210 nM T95913 CDJ10M 134142931 IC50 = 1230 nM T95913 CUE85S 134143151 IC50 > 50000 nM T95913 CQ9G7H 134145670 IC50 = 220 nM T95913 C6G8EJ 134146051 IC50 = 40000 nM T95913 CIPL93 134147099 IC50 = 2070 nM T95913 C8ITR3 134147904 IC50 > 50000 nM T95913 CXA3V0 134148445 IC50 = 3780 nM T95913 CXU92M 134150578 IC50 = 366 nM T95913 CG8LE2 134151667 IC50 < 10000 nM T95913 CK43EY 134152988 IC50 = 2940 nM T95913 CS2QP7 134154582 IC50 = 194 nM T95913 C2QGB3 134156160 IC50 = 978 nM T95913 C42RJH 134157534 IC50 = 5859 nM T95913 C9C3XT 134163708 IC50 = 0.631 nM T95913 CD9ZR6 134372929 IC50 = 440 nM T95913 CCS6I3 134372959 IC50 = 4156 nM T95913 CTD03Q 134611885 IC50 >= 199.53 nM T95913 CJXA12 134611894 IC50 <= 0.7943 nM T95913 CX0UR7 134694318 IC50 > 1000 nM T95913 C6LYD2 135121892 IC50 = 63.1 nM T95913 C9FUK2 135151360 IC50 = 52 nM T95913 CT0GQ6 135197577 IC50 = 1.7 nM T95913 C87VKA 135197594 IC50 = 0.93 nM T95913 C0YK5W 135197617 IC50 = 1.6 nM T95913 CF6DJ2 135197621 IC50 = 2.1 nM T95913 CDT25A 135197623 IC50 = 1.5 nM T95913 CQXS07 135197635 IC50 = 1.2 nM T95913 C7KXF1 135197643 IC50 = 1.3 nM T95913 CY38TL 135391000 IC50 = 89.7 nM T95913 COG86Z 135397763 IC50 = 3162.28 nM T95913 CWL67T 135397764 IC50 = 1000 nM T95913 CX8AI4 135398491 IC50 = 180 nM T95913 CQN49C 135409495 IC50 = 4000 nM T95913 C6AZ2R 135435018 IC50 > 25118.86 nM T95913 CMGY62 135485500 IC50 = 273 nM T95913 CM9NV6 135492341 IC50 = 1200 nM T95913 CWJQ64 135492555 IC50 = 968 nM T95913 C3QJ8W 135566371 IC50 = 20 nM T95913 C24ZGX 135566644 IC50 > 10000 nM T95913 C2QDV5 135566741 IC50 > 10000 nM T95913 CTJ6B2 135610083 IC50 = 5900 nM T95913 CN2ME4 135610084 IC50 = 4700 nM T95913 C4G6JF 135610087 IC50 = 5100 nM T95913 CPV59N 135685787 Ki = 1000 nM T95913 C2UN0D 135742360 IC50 > 83300 nM T95913 CI98OY 135750190 IC50 = 195 nM T95913 CF0VL3 135750206 IC50 = 48000 nM T95913 CY4CZ0 135750219 IC50 = 1300 nM T95913 CU29YK 135750268 IC50 = 680 nM T95913 C02PHA 135927892 IC50 > 25118.86 nM T95913 CS8T3D 135927897 IC50 = 5011.87 nM T95913 CF1PS8 135934877 Ki = 1300 nM T95913 C12UDA 135947972 IC50 = 187 nM T95913 CN42ZS 135947973 IC50 = 1500 nM T95913 CF8AO3 135947974 IC50 = 118 nM T95913 CW08GJ 135947976 IC50 = 89 nM T95913 C8O9HG 135947977 IC50 = 50000 nM T95913 CJN7E2 135947978 IC50 = 190 nM T95913 CFKH34 135947979 IC50 = 587 nM T95913 C58FHM 135961523 IC50 = 6918.31 nM T95913 CTRL59 135976660 Ki = 540 nM T95913 C9OAV5 135986100 IC50 = 100000 nM T95913 C3USL8 135986101 IC50 > 100000 nM T95913 C4G2HP 135995897 IC50 = 5780 nM T95913 CNF15Q 135995898 IC50 = 1340 nM T95913 C98HZG 135995899 IC50 = 7640 nM T95913 CIQ82W 135995900 IC50 = 4560 nM T95913 CP1US5 136041737 IC50 = 7070 nM T95913 CXH63V 136041747 IC50 > 10000 nM T95913 C6B5TC 136041748 IC50 > 10000 nM T95913 CU6XG1 136041749 IC50 > 10000 nM T95913 C0U5DB 136041750 IC50 > 10000 nM T95913 C48KAQ 136041752 IC50 > 10000 nM T95913 C74PRL 136041753 IC50 > 10000 nM T95913 CT4FJ1 136041757 IC50 = 10000 nM T95913 CCS2G6 136041761 IC50 > 10000 nM T95913 CEZP21 136041762 IC50 > 10000 nM T95913 CJ58TD 136041764 IC50 > 10000 nM T95913 CX67QW 136041765 IC50 > 10000 nM T95913 CK0H2Q 136041766 IC50 > 10000 nM T95913 CQP7B6 136041767 IC50 > 10000 nM T95913 CM65BS 136041773 IC50 = 8270 nM T95913 C6P7JB 136041775 IC50 > 10000 nM T95913 C5CJF7 136041776 IC50 > 10000 nM T95913 C3XIZ8 136041777 IC50 > 10000 nM T95913 C32LKO 136041785 IC50 > 10000 nM T95913 C90ARP 136041787 IC50 > 10000 nM T95913 CZ3BN1 136041792 IC50 = 6215 nM T95913 CG19DI 136041799 IC50 > 10000 nM T95913 CXJA29 136041804 IC50 = 10000 nM T95913 CHT31V 136041805 IC50 = 1590 nM T95913 CO8C4J 136041817 IC50 = 3315 nM T95913 C4QU6G 136041827 IC50 = 10000 nM T95913 CNE10X 136041834 IC50 = 10000 nM T95913 CS3AE1 136041847 IC50 > 10000 nM T95913 CZC47Y 136041848 IC50 > 10000 nM T95913 C7PHA5 136044403 IC50 = 60 nM T95913 CLA3C2 136068720 IC50 = 96.5 nM T95913 CA91JG 136069599 IC50 = 1532 nM T95913 CGAB91 136069600 IC50 = 7418 nM T95913 C3ZAW2 136069605 IC50 = 8400 nM T95913 C8JXL5 136069609 IC50 = 1000 nM T95913 C9I0EQ 136069610 IC50 = 8966 nM T95913 C25EYJ 136069611 IC50 = 2461 nM T95913 C2S5QF 136069615 IC50 = 10000 nM T95913 CI1LY8 136096349 IC50 = 60 nM T95913 CC4UM3 136176116 IC50 > 10000 nM T95913 CJRK81 136176117 IC50 > 10000 nM T95913 C63IOS 136176118 IC50 > 10000 nM T95913 C3KW7H 136176119 IC50 > 10000 nM T95913 C69AKQ 136176120 IC50 > 10000 nM T95913 CF17KO 136176121 IC50 > 10000 nM T95913 CU3TE0 136176122 IC50 = 3333 nM T95913 C3X5KE 136176124 IC50 > 10000 nM T95913 CA8C5E 136176125 IC50 > 10000 nM T95913 C5OMG2 136176126 IC50 > 10000 nM T95913 CP2YM7 136176127 IC50 > 10000 nM T95913 C8XIJ0 136176128 IC50 = 5742 nM T95913 CUY8N4 136176129 IC50 > 10000 nM T95913 C3J4ME 136176130 IC50 > 10000 nM T95913 CR1NZ2 136176131 IC50 > 10000 nM T95913 C4WG2F 136176132 IC50 > 10000 nM T95913 CJ8EC5 136176139 IC50 > 10000 nM T95913 CQ84IZ 136180335 Ki > 4000 nM T95913 C1LK9U 136183381 IC50 = 3975 nM T95913 C27TKQ 136196449 IC50 = 10000 nM T95913 CHF3R5 136200721 IC50 = 4810 nM T95913 CV2X9O 136200837 IC50 = 3690 nM T95913 CK9S4X 136229137 IC50 = 18500 nM T95913 C7S1YJ 136230225 IC50 > 10000 nM T95913 C3Q6ED 136230226 IC50 > 10000 nM T95913 CKPF02 136230227 IC50 > 10000 nM T95913 CZY9O0 136230228 IC50 = 5090 nM T95913 CRET01 136230229 IC50 > 10000 nM T95913 CX1KI8 136230230 IC50 > 10000 nM T95913 C3Z5MH 136230231 IC50 > 10000 nM T95913 CUE6N8 136230232 IC50 = 8010 nM T95913 C8Q1AP 136230233 IC50 = 6710 nM T95913 C70RXE 136230234 IC50 > 10000 nM T95913 C4W0KN 136230235 IC50 = 6610 nM T95913 CMZN01 136230236 IC50 > 10000 nM T95913 CCU0H5 136241428 IC50 = 1780 nM T95913 C75RWX 136244223 IC50 = 7410 nM T95913 CXI04C 136244224 IC50 = 6480 nM T95913 C0YW6L 136244283 IC50 = 1340 nM T95913 CF3DK1 136245085 IC50 = 9360 nM T95913 CEU87Z 136245089 IC50 = 10000 nM T95913 CUF56H 136245251 IC50 = 2170 nM T95913 CKPR81 136245252 IC50 = 7120 nM T95913 C7C5ZV 136249323 IC50 = 2600 nM T95913 CI6HG4 136249373 IC50 = 264 nM T95913 CL4MO3 136249382 IC50 = 10000 nM T95913 C68CRX 136254271 IC50 = 2870 nM T95913 C0GZV9 136254283 IC50 > 10000 nM T95913 CMWA86 136264282 IC50 = 9149 nM T95913 CSD78N 136264452 IC50 = 6390 nM T95913 C1HI5T 136264454 IC50 = 1131 nM T95913 CV3UE9 137333450 IC50 = 202.7 nM T95913 CH8WU5 137348751 IC50 = 12.59 nM T95913 CP34TI 137631388 IC50 = 130 nM T95913 CF0PQ2 137632018 IC50 > 794.33 nM T95913 CZ4WN6 137633048 Ki = 66.7 nM T95913 CIX4S7 137633081 IC50 = 630.96 nM T95913 CR17XH 137634463 IC50 = 499 nM T95913 CM63EP 137634801 IC50 = 6309.57 nM T95913 CYAL31 137634808 Ki = 113 nM T95913 C34MHP 137634951 IC50 = 35 nM T95913 C9GXM1 137635017 IC50 = 794.33 nM T95913 C06BDR 137635072 IC50 = 150 nM T95913 CY86AJ 137635564 IC50 = 630.96 nM T95913 CYK6C4 137635941 IC50 >= 199.53 nM T95913 CMN6T7 137636115 IC50 = 125 nM T95913 CZ74XF 137636132 IC50 = 316.23 nM T95913 CPJ43Y 137636841 IC50 = 220 nM T95913 C7BE2O 137636964 IC50 = 10000 nM T95913 CV38QX 137637076 IC50 > 1000 nM T95913 CK4V7A 137637244 IC50 = 2511.89 nM T95913 CK2HR6 137637299 IC50 = 4300 nM T95913 CXPI97 137637422 IC50 >= 199.53 nM T95913 CX8NI0 137637899 IC50 = 15848.93 nM T95913 CMZV19 137639099 IC50 = 199.53 nM T95913 CJ3LX4 137639119 IC50 = 4.7 nM T95913 CS78JW 137639139 IC50 = 43 nM T95913 CHK7G9 137639570 IC50 = 6309.57 nM T95913 C4TSZ8 137639858 IC50 = 316.23 nM T95913 CK9GP8 137640140 Ki > 490 nM T95913 C7HA4V 137640279 IC50 >= 199.53 nM T95913 CA0QO6 137640453 IC50 = 91.9 nM T95913 CWK2F4 137640548 IC50 > 31622.78 nM T95913 C67NLM 137640896 IC50 >= 199.53 nM T95913 CQ8X0E 137641383 IC50 = 99 nM T95913 C0I6RQ 137641405 IC50 = 1000 nM T95913 CN3F5A 137641753 IC50 >= 199.53 nM T95913 C5X3TH 137642662 IC50 = 27 nM T95913 C1EBS6 137642764 Ki > 490 nM T95913 C8M9TX 137642801 IC50 = 16 nM T95913 CL4Q9G 137643238 IC50 > 1000 nM T95913 CP3JK1 137643598 IC50 = 794.33 nM T95913 CAPQ93 137644458 IC50 = 251.19 nM T95913 C4KAU7 137644907 IC50 = 7943.28 nM T95913 CKI2G8 137645541 IC50 = 398.11 nM T95913 C6SW7U 137646075 IC50 >= 199.53 nM T95913 C9SU6F 137646331 IC50 = 630.96 nM T95913 C5ERV3 137646413 IC50 = 29 nM T95913 CZC27Y 137646667 IC50 = 158.49 nM T95913 CA4V8H 137646998 IC50 >= 199.53 nM T95913 C5HIM9 137647114 IC50 = 398.11 nM T95913 CPMG65 137647250 IC50 = 8.4 nM T95913 C3TXN9 137647591 IC50 = 291 nM T95913 CPX42N 137647765 IC50 = 190 nM T95913 C6OK0J 137647964 IC50 > 19952.62 nM T95913 CS39XP 137648085 IC50 = 251.19 nM T95913 C4Z0NQ 137648826 IC50 = 1584.89 nM T95913 CE54DO 137648917 IC50 >= 199.53 nM T95913 CSML14 137649696 IC50 = 47 nM T95913 CCM18K 137650283 IC50 = 794.33 nM T95913 CHT1R8 137650579 IC50 = 794.33 nM T95913 C9QA0W 137652944 IC50 >= 199.53 nM T95913 CI64CW 137653468 IC50 > 25118.86 nM T95913 CN78RE 137653565 IC50 = 501.19 nM T95913 CTKQ38 137653713 IC50 = 199.53 nM T95913 C9M4PI 137653924 IC50 = 398.11 nM T95913 C9E5JK 137654836 IC50 = 316.23 nM T95913 CD19ZS 137654937 IC50 = 61 nM T95913 C4N5LS 137655123 IC50 = 1000 nM T95913 C82EOF 137655140 IC50 = 316.23 nM T95913 CHV26G 137655828 IC50 = 20 nM T95913 CC5NK4 137655965 IC50 = 501.19 nM T95913 CLC7N4 137656507 IC50 = 630.96 nM T95913 CE9H8D 137657006 IC50 = 1995.26 nM T95913 C3TD6A 137657429 Ki = 84.3 nM T95913 C2JX1W 137657572 IC50 >= 199.53 nM T95913 C41OPW 137658031 IC50 = 3162.28 nM T95913 C6BF8E 137658458 IC50 = 390 nM T95913 C35DPY 137658611 IC50 = 398.11 nM T95913 CU9PB7 137659393 IC50 = 501.19 nM T95913 CZ36BW 137659557 IC50 = 501.19 nM T95913 C3CF4O 137659746 IC50 = 316.23 nM T95913 CCX64Q 137660055 IC50 = 398.11 nM T95913 C1F6QN 137660818 IC50 >= 199.53 nM T95913 CP5K4E 137660883 IC50 = 132 nM T95913 C1OLQ3 137660961 IC50 = 1258.93 nM T95913 CM6FS2 137661095 IC50 = 398.11 nM T95913 C8R3JK 137661301 IC50 = 158.49 nM T95913 C9HPG8 137661516 IC50 = 1584.89 nM T95913 C90ELH 137661890 IC50 = 187 nM T95913 CA3C4O 138454792 IC50 = 67 nM T95913 CKDZ26 138504497 IC50 = 2900 nM T95913 C0BFS3 139327957 IC50 = 140 nM T95913 C7ZAQ1 141406387 IC50 = 24640 nM T95913 C7NUI8 141406388 IC50 = 42570 nM T95913 CQYI18 141406390 IC50 = 9470 nM T95913 CUA1D0 141406392 IC50 = 38290 nM T95913 CP0R6Y 141406393 IC50 = 1900 nM T95913 C1EVQ0 141406394 IC50 = 17810 nM T95913 C2QP0F 141406396 IC50 = 18240 nM T95913 CY2M0B 141406399 IC50 = 5100 nM T95913 CC3OU2 141406400 IC50 = 32180 nM T95913 CKV13Y 141406404 IC50 = 19030 nM T95913 C3Q1VL 141419885 IC50 = 174.2 nM T95913 C3EJX8 141419888 IC50 = 198.5 nM T95913 CKX4P3 141446054 IC50 > 158489.32 nM T95913 C9IV8R 141461655 IC50 = 268 nM T95913 C4C0QL 141461656 IC50 = 37 nM T95913 CG6O8P 141461658 IC50 = 63 nM T95913 C6I1VW 141461659 IC50 = 155 nM T95913 CES84U 141461662 IC50 = 1593 nM T95913 CM8HT7 141461664 IC50 = 381 nM T95913 CZV17F 141461667 IC50 = 7 nM T95913 CFR0I4 141461668 IC50 = 2062 nM T95913 CD5VE0 141461669 IC50 = 17 nM T95913 CU6LE4 141461671 IC50 = 15 nM T95913 CHJ93Y 141461672 IC50 = 2966 nM T95913 CV54CS 141471198 IC50 = 11 nM T95913 C25HYI 141471200 IC50 = 10 nM T95913 CZS03J 141509623 IC50 = 684 nM T95913 C1R9AN 141518981 IC50 = 45 nM T95913 C4MH5U 141518989 IC50 = 37 nM T95913 CQT27N 141520958 IC50 = 116 nM T95913 CH5F2X 141716982 IC50 = 1.259 nM T95913 CRU08D 141717009 IC50 = 0.7943 nM T95913 C8Q0VB 141717016 IC50 = 1.259 nM T95913 CQ34YR 142506035 IC50 = 162 nM T95913 CU03GW 142506036 IC50 = 2 nM T95913 C74MXW 142506065 IC50 = 3 nM T95913 CX6BQ7 142506102 IC50 = 2 nM T95913 CY3BM0 142506119 IC50 = 1769 nM T95913 CC6MD0 142506155 IC50 = 8 nM T95913 C05QOM 142506157 IC50 = 203 nM T95913 CGNQ74 142506189 IC50 = 103 nM T95913 CT3U9R 142506192 IC50 = 2 nM T95913 C1T3IQ 142506210 IC50 = 43 nM T95913 CEGV67 142506220 IC50 = 234 nM T95913 CP5HF8 142506225 IC50 = 995 nM T95913 C1U3CA 142506238 IC50 = 45 nM T95913 C7QMG9 145108300 IC50 = 17 nM T95913 C1FIE4 145439085 IC50 = 2293 nM T95913 CGF4I3 145946093 IC50 = 316.23 nM T95913 CI40JE 145951013 IC50 = 602.1 nM T95913 C6YT8E 145951131 IC50 > 9100 nM T95913 CFW62M 145951569 IC50 = 120.5 nM T95913 CHA84K 145951830 IC50 > 10000 nM T95913 CT4I9A 145952160 IC50 = 31 nM T95913 C91GVH 145952598 IC50 = 76 nM T95913 C1W0GJ 145952796 IC50 = 25118.86 nM T95913 CVMF13 145953272 IC50 = 1207 nM T95913 CYL5T1 145953372 IC50 <= 10000 nM T95913 CP14AV 145953653 IC50 = 751 nM T95913 CY8D5Q 145953886 IC50 = 596.3 nM T95913 C3ZUW8 145954195 IC50 = 358.3 nM T95913 C1NJB7 145955070 IC50 = 47 nM T95913 CRHE01 145955133 IC50 <= 10000 nM T95913 C7MP9Z 145955279 IC50 = 255.7 nM T95913 C7K8VT 145955565 IC50 = 118.1 nM T95913 CPU4X2 145955670 IC50 = 1898 nM T95913 C3ST5Y 145955693 IC50 = 140 nM T95913 C1VH5X 145955836 IC50 = 2628 nM T95913 C7K2YF 145956631 IC50 <= 10000 nM T95913 CQW74M 145956683 IC50 = 110 nM T95913 CJ1F6A 145956725 IC50 = 1036 nM T95913 C12IFO 145956886 IC50 = 456.7 nM T95913 C9O2PL 145958063 IC50 = 193.7 nM T95913 CQH01X 145958257 IC50 <= 10000 nM T95913 C3DGU7 145958571 IC50 = 708 nM T95913 C9NS6T 145958690 IC50 = 245.5 nM T95913 C7ZO9V 145959196 IC50 = 236 nM T95913 CSC81H 145959429 IC50 = 62 nM T95913 C0S1YM 145959980 IC50 = 303 nM T95913 CT3I2R 145960112 IC50 = 893.1 nM T95913 C8MJ9X 145960272 IC50 = 170 nM T95913 CLH5J2 145960703 IC50 = 6.31 nM T95913 CF36RA 145961004 IC50 = 64 nM T95913 CZO6T7 145961089 IC50 = 2511.89 nM T95913 CX6T3J 145961172 IC50 > 10000 nM T95913 C9I7EC 145961182 IC50 = 7.943 nM T95913 C54ZQA 145961234 IC50 = 3981.07 nM T95913 C83FPK 145961240 IC50 = 100 nM T95913 C31QBE 145961348 IC50 > 10000 nM T95913 CHF56O 145961403 IC50 > 9100 nM T95913 C2GT9Y 145961404 IC50 > 9100 nM T95913 COCG81 145961565 IC50 = 6309.57 nM T95913 C73MVW 145961583 IC50 = 1584.89 nM T95913 CKF0I1 145961740 IC50 = 1.259 nM T95913 C6HB9M 145961899 IC50 = 6309.57 nM T95913 CS46RM 145962397 Ki = 160 nM T95913 CT42OW 145962848 IC50 = 25.12 nM T95913 CLFQ85 145963006 IC50 = 12.59 nM T95913 CAI0D6 145963117 IC50 = 256 nM T95913 CA4FO3 145963201 IC50 = 10 nM T95913 CYZ14S 145963250 IC50 = 7943.28 nM T95913 CAD5Q9 145963302 IC50 > 10000 nM T95913 C35ZRP 145963416 IC50 > 10000 nM T95913 CQBU31 145963478 IC50 > 1000 nM T95913 C0S1ZI 145963484 IC50 = 1.259 nM T95913 C4JI8B 145963558 IC50 = 158.49 nM T95913 C87HFG 145964719 IC50 = 4752 nM T95913 CRE3Q1 145966313 IC50 = 68 nM T95913 CU9XC4 145966764 IC50 = 0.7 nM T95913 C97IKW 145969580 IC50 = 223.9 nM T95913 CK82QG 145969816 IC50 = 1783 nM T95913 C71YAK 145970017 IC50 = 3000 nM T95913 C3Y7RS 145970202 IC50 > 10000 nM T95913 CP6YC2 145970436 IC50 = 117.5 nM T95913 CZ98FH 145971490 IC50 = 1591 nM T95913 CTB97Z 145971948 IC50 = 408 nM T95913 CGQJ04 145972017 IC50 = 1590 nM T95913 C96IUM 145973569 IC50 = 0.5 nM T95913 CD7PS3 145973794 IC50 = 420 nM T95913 CZ9G6E 145974533 IC50 = 146 nM T95913 C3XIT8 145974725 IC50 = 1491 nM T95913 C1N5TZ 145975623 IC50 = 445 nM T95913 C3LR4O 145976442 IC50 = 3560 nM T95913 C3YG4Z 145977475 IC50 = 0.7 nM T95913 CPZS56 145982349 EC50 = 10000 nM T95913 CH90CT 145983168 IC50 = 184.7 nM T95913 CJU02I 145983624 IC50 = 62 nM T95913 CVS2U0 145983808 IC50 = 363 nM T95913 CF8MR5 145986347 IC50 = 1000 nM T95913 C6XMQ8 145989163 EC50 = 9890 nM T95913 CBU86Y 145991850 IC50 = 10000 nM T95913 C8X2IT 145996536 IC50 > 10000 nM T95913 C4K0JW 145996540 IC50 = 1.2 nM T95913 C6RPG0 146014481 IC50 = 831.76 nM T95913 C59KOM 146585662 IC50 = 9 nM T95913 CFQO97 146585699 IC50 = 752 nM T95913 C0GMR1 146585718 IC50 = 135 nM T95913 CI85VS 146731761 IC50 = 81 nM T95913 CWZ05D 148564044 IC50 = 22 nM T95913 C4MC0S 149169124 IC50 = 1870 nM T95913 CVW62P 149242889 IC50 = 10530 nM T95913 CN87RZ 149370890 IC50 = 810 nM T95913 CK4FJ1 149556361 IC50 = 2300 nM T95913 C8UQL4 153940691 IC50 = 1320 nM T95913 CMZ68Q 153940692 IC50 = 110 nM T95913 C5X7JK 154734328 IC50 = 1000 nM T95913 C8Q9UG 155510876 IC50 = 222 nM T95913 CDT8F2 155510913 IC50 = 1258.93 nM T95913 C6WIC9 155511977 IC50 = 1258.93 nM T95913 CPH8N1 155512095 IC50 = 251.19 nM T95913 CZJ9D6 155512258 IC50 = 5533 nM T95913 CG9I4X 155512515 IC50 = 140 nM T95913 CR1Z8A 155512529 IC50 > 10000 nM T95913 CQZY50 155512775 IC50 = 39.81 nM T95913 C5V2GO 155512947 IC50 = 2511.89 nM T95913 C1DIT4 155513047 IC50 = 125.89 nM T95913 C8PG6Z 155513084 IC50 = 794.33 nM T95913 C5M6NS 155513226 IC50 = 9550 nM T95913 C45SYX 155513615 IC50 = 6 nM T95913 CBH57O 155514764 IC50 = 2511.89 nM T95913 C5C9EG 155515047 IC50 = 1000 nM T95913 CEFS61 155515135 IC50 = 2650 nM T95913 C0AXF7 155515394 IC50 = 1584.89 nM T95913 CTS48F 155515676 IC50 = 3 nM T95913 C7Q3FR 155515734 IC50 = 1995.26 nM T95913 C30ZFN 155516445 IC50 = 630.96 nM T95913 CJDG04 155516604 IC50 = 100 nM T95913 C42JXQ 155517064 IC50 = 1995.26 nM T95913 CYO19V 155517071 IC50 = 125.89 nM T95913 CYWX76 155517213 IC50 = 1584.89 nM T95913 CT53XD 155517442 IC50 = 12589.25 nM T95913 C4G8YN 155517534 IC50 = 1983 nM T95913 CS2JT9 155518175 IC50 = 3162.28 nM T95913 CW7OM6 155518918 IC50 = 708 nM T95913 CC51GM 155519635 IC50 = 158.49 nM T95913 CHFJ25 155519726 IC50 = 12589.25 nM T95913 CZ78HW 155519830 IC50 = 316.23 nM T95913 CQEK39 155520373 IC50 = 4.3 nM T95913 C3D7FJ 155520444 IC50 = 6309.57 nM T95913 C5D6YX 155521099 IC50 > 10000 nM T95913 CEA3M1 155521494 IC50 = 63.1 nM T95913 CBSR95 155522042 IC50 = 3480 nM T95913 CZO7Q8 155522149 IC50 = 536 nM T95913 CCGW06 155523124 IC50 = 6309.57 nM T95913 CNB70P 155523246 IC50 = 1000 nM T95913 C4TLQ7 155523447 IC50 > 10000 nM T95913 CZG27I 155523570 IC50 = 38 nM T95913 C37RVF 155523599 IC50 = 4500 nM T95913 C4H2AB 155524238 IC50 = 15.85 nM T95913 CP18VT 155524467 IC50 = 1995.26 nM T95913 CUP7L2 155524901 IC50 = 1258.93 nM T95913 C2BL5I 155525312 IC50 = 25.12 nM T95913 C10RZQ 155525477 IC50 = 1000 nM T95913 CF76OV 155525717 IC50 = 19.3 nM T95913 C0UA4D 155525996 IC50 = 63.1 nM T95913 C0AR4W 155526097 IC50 = 3981.07 nM T95913 C3EAR8 155526323 IC50 = 1000 nM T95913 C82NUW 155527501 IC50 = 445 nM T95913 CK07GS 155527559 IC50 = 64 nM T95913 CX12MK 155527651 IC50 = 4 nM T95913 C8Z3TK 155528581 IC50 = 1584.89 nM T95913 C0B2NV 155528644 IC50 = 853 nM T95913 C3VAI9 155528997 IC50 = 501.19 nM T95913 C9L6OC 155529247 IC50 = 467 nM T95913 C2FE1S 155529479 IC50 = 25.12 nM T95913 CB90AR 155529643 IC50 = 199.53 nM T95913 CFV1S0 155529706 IC50 = 434 nM T95913 C14QOF 155530163 IC50 = 1584.89 nM T95913 C4I5UP 155530224 IC50 = 158.49 nM T95913 CX6N3Y 155531155 IC50 = 79.43 nM T95913 C9AXO7 155531257 IC50 = 1258.93 nM T95913 CGAI60 155531409 IC50 = 3162.28 nM T95913 CDI4V8 155531526 IC50 = 194 nM T95913 CE6QP1 155532037 IC50 = 501.19 nM T95913 CJH9U4 155532237 IC50 = 12589.25 nM T95913 C6W0JX 155532471 IC50 = 6309.57 nM T95913 CKMD29 155532546 IC50 = 6309.57 nM T95913 C3XFB8 155532820 IC50 = 19.95 nM T95913 CIYA39 155532858 IC50 = 34 nM T95913 C0GR1J 155533050 IC50 = 2 nM T95913 CQS8P1 155533070 IC50 = 1584.89 nM T95913 C0SZR9 155533335 IC50 = 2511.89 nM T95913 CAT9V1 155533370 IC50 = 5600 nM T95913 C67ERP 155533384 IC50 = 158.49 nM T95913 CL8OM7 155533564 IC50 = 6081 nM T95913 CBM24U 155533579 IC50 = 3981.07 nM T95913 CR5H8B 155533591 IC50 = 1995.26 nM T95913 CA7T0Y 155533911 IC50 = 9340 nM T95913 C8XQ4W 155534168 IC50 = 87 nM T95913 CN1ST4 155534269 IC50 = 1258.93 nM T95913 CBEG39 155534594 IC50 = 1258.93 nM T95913 CTZ3E0 155534905 IC50 = 112 nM T95913 CG1JR7 155535513 IC50 = 630.96 nM T95913 CN6KJ5 155535520 IC50 = 794.33 nM T95913 C5F2TY 155535537 IC50 = 1995.26 nM T95913 CKB2U4 155535691 IC50 = 63.1 nM T95913 CY7X3M 155535740 IC50 = 39.81 nM T95913 CUWE49 155535963 IC50 = 794.33 nM T95913 C70UDF 155536179 IC50 = 3162.28 nM T95913 CEJ6L1 155536226 IC50 = 210.7 nM T95913 CNB24M 155536473 IC50 = 1000 nM T95913 C2CG1A 155537016 IC50 = 3981.07 nM T95913 C8AJ6C 155538256 IC50 = 250.4 nM T95913 CQ1E6H 155538266 IC50 = 39.81 nM T95913 CZ19AN 155538609 IC50 = 496 nM T95913 CHR8M1 155538990 IC50 = 7510 nM T95913 CC1BG2 155539321 IC50 > 10000 nM T95913 CF20PS 155539394 IC50 = 2511.89 nM T95913 C8LKW4 155540264 IC50 = 2511.89 nM T95913 C6I5DK 155541290 IC50 = 1258.93 nM T95913 CECX47 155541544 IC50 = 501.19 nM T95913 C4FC0V 155541900 IC50 = 630.96 nM T95913 CKBW37 155542030 IC50 = 1905 nM T95913 CASE16 155542363 IC50 = 3162.28 nM T95913 C8AXF9 155542633 IC50 = 5011.87 nM T95913 C8OC2P 155542800 IC50 = 5600 nM T95913 C42BIZ 155542813 IC50 = 12589.25 nM T95913 CVNR95 155542898 IC50 = 1400 nM T95913 C1SY0G 155543154 IC50 = 23200 nM T95913 C7IWJ2 155543389 IC50 = 10000 nM T95913 CZY0N4 155543588 IC50 = 10 nM T95913 CJB8C9 155543659 IC50 = 231 nM T95913 CX1C8I 155544561 IC50 > 10000 nM T95913 CBN29V 155544583 IC50 = 204 nM T95913 C98FXC 155544955 IC50 = 3594 nM T95913 CTSW53 155546042 IC50 > 10000 nM T95913 CQ6J7U 155546361 IC50 = 280 nM T95913 C8SQA2 155546999 IC50 = 12.59 nM T95913 C8D4ZH 155547166 IC50 = 630.96 nM T95913 CI6KO7 155548518 IC50 = 251.19 nM T95913 CL4F8P 155549003 IC50 = 7.943 nM T95913 CM6S8K 155549098 IC50 = 5011.87 nM T95913 C4PEJ5 155549895 IC50 > 10000 nM T95913 CFP94J 155550309 IC50 = 794.33 nM T95913 CQ5OD0 155550395 IC50 = 45 nM T95913 CK1JR7 155551961 IC50 = 6.5 nM T95913 CJ75BO 155552100 IC50 > 1000 nM T95913 CXN3Y8 155553327 IC50 = 3981.07 nM T95913 CL04BD 155554125 IC50 = 934 nM T95913 CX9C6O 155554180 IC50 = 1000 nM T95913 CC13QL 155555170 IC50 = 1378 nM T95913 CZX06J 155555458 IC50 = 1995.26 nM T95913 C2OGW1 155555483 IC50 = 521 nM T95913 CRO5Z3 155556073 IC50 = 5756 nM T95913 CH2P4T 155556124 IC50 = 25118.86 nM T95913 CCU8M1 155556480 IC50 = 15848.93 nM T95913 CIU29Z 155556576 IC50 > 10000 nM T95913 CM3LI6 155556593 IC50 > 10000 nM T95913 CZ8CX1 155556887 IC50 = 501.19 nM T95913 CG2FS6 155557123 IC50 = 2511.89 nM T95913 CFS63H 155557182 IC50 = 301 nM T95913 C0FE4G 155557988 IC50 = 2183 nM T95913 CR8J0E 155558167 IC50 = 50.12 nM T95913 CN96JH 155558197 IC50 = 316.23 nM T95913 CSO4M3 155558261 IC50 = 5011.87 nM T95913 C52TSP 155558262 IC50 = 440 nM T95913 CS70ER 155559192 IC50 = 247 nM T95913 CVG49I 155560688 IC50 = 4010 nM T95913 C5S7AL 155560766 IC50 = 199.53 nM T95913 CQ7PS9 155560780 IC50 = 3981.07 nM T95913 CLO3B1 155561152 IC50 = 7900 nM T95913 C8XS0L 155561165 IC50 = 794.33 nM T95913 C72CQG 155561233 IC50 = 125.89 nM T95913 C1INL7 155561328 IC50 = 794.33 nM T95913 CX6U2T 155562388 IC50 = 3981.07 nM T95913 C5E9TP 155562641 IC50 = 79432.82 nM T95913 CCF4W2 155563986 IC50 = 6309.57 nM T95913 CHK4E8 155565269 IC50 = 1258.93 nM T95913 C7PXA0 155565551 IC50 = 630.96 nM T95913 CY4N7O 155565715 IC50 = 15848.93 nM T95913 CVQ6Z4 155565763 IC50 = 2511.89 nM T95913 CA1RX3 155565771 IC50 = 2511.89 nM T95913 CQ3AU4 155565828 IC50 = 19952.62 nM T95913 CMK4I3 155565845 IC50 = 1995.26 nM T95913 C59VPW 155565958 IC50 = 1584.89 nM T95913 CAP9F2 155566187 IC50 = 15 nM T95913 CM7E2G 155566279 IC50 = 3162.28 nM T95913 C3BNY5 155566309 IC50 = 10000 nM T95913 C9KQW3 155567372 IC50 = 740 nM T95913 C98NZE 155567616 IC50 = 5011.87 nM T95913 C1HQ5J 155568324 IC50 = 354 nM T95913 CLA46O 155568356 IC50 = 800 nM T95913 C7SLR8 155568452 IC50 = 501.19 nM T95913 C1S8ZB 155568922 IC50 > 1000 nM T95913 C14LVO 155569074 IC50 = 158.49 nM T95913 CFWP17 155569113 IC50 = 587 nM T95913 CUH38L 155569363 IC50 = 8420 nM T95913 C4H0NE 155569598 IC50 = 3162.28 nM T95913 D00GQM 25069592 IC50 = 7972 nM T95913 D00ZIK 9908783 IC50 = 61000 nM T95913 D01ILN 223355 IC50 = 8500 nM T95913 D01SSI 24937012 IC50 > 10000 nM T95913 D03EHM 24905142 IC50 = 1100 nM T95913 D03QQH 16760391 IC50 = 100000 nM T95913 D05USL 5278396 IC50 > 1000 nM T95913 D06DNH 9907093 IC50 > 10000 nM T95913 D06HVH 54613583 IC50 = 3100 nM T95913 D06PWI 42623951 IC50 = 25.12 nM T95913 D07JKB 135955185 IC50 = 5135 nM T95913 D07PMP 44187953 IC50 = 16 nM T95913 D08KSQ 11637090 IC50 > 10000 nM T95913 D08NQM 5289247 IC50 = 8 nM T95913 D09FBN 135955186 IC50 = 8558 nM T95913 D09ZNV 447682 IC50 > 200000 nM T95913 D0AH8Q 25074311 IC50 = 6742 nM T95913 D0EU1R 46215815 IC50 = 25118 nM T95913 D0F1SI 25074312 IC50 = 8000 nM T95913 D0H0HR 49836027 IC50 = 171 nM T95913 D0H2CM 135565635 IC50 = 1300 nM T95913 D0P5TI 58441401 IC50 = 240.3 nM T95913 D0R0TW 11964036 IC50 = 590 nM T95913 D0R2UG 52936849 IC50 = 104 nM T95913 D0S5YV 6852167 Ki = 7 nM T95913 D0T3PW 5281672 IC50 = 4720 nM T95913 D0TC5H 16049458 IC50 = 2343 nM T95913 D0W8XH 9884685 IC50 = 15 nM T95913 D0Y1DR 46225260 IC50 = 7371 nM T95913 D0Y3OO 11327430 IC50 = 220 nM T66011 CM86EA 25082538 IC50 = 12000 nM T66011 C8J7CH 44560082 IC50 = 19000 nM T66011 C2GXT8 44560086 IC50 = 19000 nM T66011 CA03BN 46883572 IC50 = 19000 nM T66011 CV0W3Y 46883575 IC50 = 23000 nM T66011 C8R2WL 46883576 IC50 = 13000 nM T66011 CGFC59 46883582 IC50 = 4000 nM T66011 C87DPG 46883583 IC50 = 5000 nM T66011 CR51BY 46883590 IC50 = 5000 nM T66011 CKA62U 46883591 IC50 = 12000 nM T66011 C5Z7YU 46883592 IC50 = 3000 nM T66011 CHWU39 46883593 IC50 = 3000 nM T66011 C1SB3M 46883594 IC50 = 50000 nM T66011 CC6SH3 46883595 IC50 = 7000 nM T66011 C14TGE 86282201 IC50 = 30 nM T66011 C5T3ZX 91755031 IC50 = 23 nM T66011 CVMB75 118046356 IC50 = 1 nM T66011 CL74ZP 145985971 IC50 = 250 nM T66011 D09JGO 46883596 IC50 = 10000 nM T16016 D0I1FQ 54671008 Ki = 5 nM T16016 D00XBC 46861584 IC50 > 10000 nM T16016 D05VTN 135565361 IC50 = 2 nM T16016 D0O2XQ 11256587 IC50 > 10000 nM T16016 D0UX2V 44537841 IC50 = 1.5 nM T16016 D0W0LS 183789 IC50 > 10000 nM T16016 C7Y8VS 1318 EC50 = 5900 nM T16016 CB4Z9P 1474 EC50 = 31622.78 nM T16016 C78GSK 14338 EC50 = 3600 nM T16016 CW6J7R 15664 EC50 = 15848.93 nM T16016 CBX47E 20445 EC50 = 12000 nM T16016 CD72TB 65237 IC50 < 1000000 nM T16016 CF1UA4 70848 EC50 = 63095.73 nM T16016 CR15FN 72791 EC50 = 1800 nM T16016 C8SC9N 72792 EC50 = 794.33 nM T16016 C7SIE4 74265 EC50 = 1500 nM T16016 CMJ4V7 77524 EC50 < 100000 nM T16016 CGZ1C6 77865 EC50 = 1995.26 nM T16016 CBW4N5 93149 EC50 = 1000 nM T16016 CTUE81 336912 IC50 > 1000000 nM T16016 C2P3FM 353741 EC50 = 15000 nM T16016 CQ3KO7 483339 IC50 > 1000 nM T16016 C7AP9W 483340 IC50 > 1000 nM T16016 CAB79M 483341 IC50 > 1000 nM T16016 C7XW2D 483342 IC50 > 1000 nM T16016 C7PMT6 483343 IC50 > 1000 nM T16016 CP25RI 483344 IC50 > 1000 nM T16016 CSF9D4 602123 IC50 = 5011.87 nM T16016 CXMY27 619353 EC50 < 1000000 nM T16016 CYU56N 667748 EC50 = 1200 nM T16016 C1SFP9 1370410 IC50 = 93 nM T16016 CAF8P7 2733927 EC50 = 10000 nM T16016 CJ73WC 2868511 Ki = 537.03 nM T16016 CAVN29 3063066 Ki = 203 nM T16016 CP65DT 3063068 Ki = 164 nM T16016 C1TX2Y 3794409 Ki = 67 nM T16016 CPZ6S1 3796276 Ki = 85.11 nM T16016 CI4N9O 3798520 Ki = 162 nM T16016 CI73AQ 5311125 Ki = 24 nM T16016 CMT8K7 5481702 IC50 = 10000 nM T16016 CHCY06 6918496 IC50 = 0.9 nM T16016 C18KRM 6918497 IC50 = 0.9 nM T16016 C5IXA6 7693048 IC50 > 10000 nM T16016 CEA5Y0 9804868 Ki = 44 nM T16016 CXM5S9 9845614 IC50 = 400 nM T16016 CUES31 9850002 Ki = 22 nM T16016 CC9U3T 9857981 Ki = 54.95 nM T16016 CN25EM 9869274 Ki = 56 nM T16016 CK7FJ6 9870185 IC50 = 5011.87 nM T16016 CK97YH 9870787 Ki = 54 nM T16016 CE13DO 9889700 Ki = 52 nM T16016 CN92IT 9894713 IC50 = 5.2 nM T16016 C2R6KA 9902204 Ki = 38.9 nM T16016 C0RH2D 9902578 Ki = 28.84 nM T16016 CY4B8U 9924108 Ki = 57 nM T16016 CQ86OZ 9935062 IC50 = 23 nM T16016 C24MLV 9935588 IC50 > 50000 nM T16016 C7LY1M 9945265 Ki = 54.95 nM T16016 C7WM0Z 9954423 IC50 = 0.96 nM T16016 C91RTG 9956238 IC50 > 10000 nM T16016 C56NZO 9956380 Ki = 45 nM T16016 CTO01C 9956488 Ki = 34 nM T16016 CAVL67 9959839 Ki = 9 nM T16016 CL3KT8 9967166 Ki = 165.96 nM T16016 CTFZ89 9967349 Ki = 27.54 nM T16016 CBVP31 9967465 Ki = 524.81 nM T16016 CJ2HT6 9979012 IC50 = 4200 nM T16016 C3TB8W 9980155 IC50 = 0.9 nM T16016 C3L7CB 9999626 IC50 = 860 nM T16016 CH5C2N 10000888 IC50 = 7100 nM T16016 CG8R5H 10001921 IC50 = 58 nM T16016 C0PDB1 10003548 IC50 = 1 nM T16016 CWD3B7 10030344 IC50 = 6.7 nM T16016 C6V8MF 10032207 IC50 = 0.92 nM T16016 C1T2FI 10049290 IC50 = 650 nM T16016 CIYE32 10049340 IC50 = 28 nM T16016 C81WKZ 10072252 IC50 = 20 nM T16016 C5QHG3 10072781 IC50 = 2.8 nM T16016 CYAJ69 10073725 IC50 = 12 nM T16016 C9RM2X 10076509 Ki = 22 nM T16016 CG0MA2 10094211 IC50 = 3.2 nM T16016 CV18TY 10094212 IC50 = 0.52 nM T16016 CC03WA 10111333 Ki = 10.47 nM T16016 CM48CP 10132885 Ki = 21.88 nM T16016 CFH9U0 10133557 Ki = 138.04 nM T16016 CU90AP 10195332 Ki = 5 nM T16016 CIGL41 10254761 IC50 = 8.9 nM T16016 CL0BS6 10255511 IC50 = 32 nM T16016 CK49NQ 10272003 IC50 > 10000 nM T16016 CDU26C 10293022 Ki = 23.99 nM T16016 CZNP37 10300214 Ki = 15.85 nM T16016 CWFB30 10323427 IC50 > 1000 nM T16016 CFH29X 10367570 IC50 = 1.4 nM T16016 C93OHM 10368175 IC50 = 1.8 nM T16016 C2JX8W 10368788 IC50 = 7.9 nM T16016 CFAY08 10371087 Ki = 1.8 nM T16016 C58GLR 10388824 IC50 = 13 nM T16016 C5LJ4B 10389562 IC50 = 0.9 nM T16016 CM9R2K 10391877 IC50 = 71 nM T16016 C9WC5D 10393066 IC50 = 3.2 nM T16016 CQU29H 10409538 IC50 = 0.96 nM T16016 C56SLV 10412648 IC50 = 1.4 nM T16016 CI9A3D 10434371 IC50 = 1.5 nM T16016 C4R6KU 10435088 IC50 = 400 nM T16016 C5GQF1 10436125 IC50 = 1.9 nM T16016 CY9B4E 10456104 IC50 = 9 nM T16016 CP1X2E 10478859 IC50 = 0.64 nM T16016 C4LB6P 10480588 IC50 = 2.5 nM T16016 CEW7C9 10482996 IC50 = 5.6 nM T16016 C6VI1Y 10499297 Ki = 54 nM T16016 C0AF4N 10501338 Ki = 306 nM T16016 CRK86P 10502989 IC50 = 1600 nM T16016 CP0OT1 10503474 Ki = 385 nM T16016 C4R5MW 10503785 Ki = 130 nM T16016 CH0F6V 10505512 IC50 = 240 nM T16016 CB6C7M 10507822 IC50 = 3.6 nM T16016 C9DY4N 10509338 IC50 = 3.1 nM T16016 C8CX5H 10524463 Ki = 4010 nM T16016 CVT27G 10525291 IC50 = 200 nM T16016 C2XON9 10525695 Ki = 906 nM T16016 CSRY03 10528677 Ki = 1330 nM T16016 CV42OK 10530837 Ki = 224 nM T16016 CIR60O 10531238 IC50 = 2100 nM T16016 CNO9H4 10531631 IC50 = 2.8 nM T16016 C4HSF7 10547456 Ki = 128 nM T16016 CUMX19 10548809 Ki = 93 nM T16016 CO6V8R 10549688 Ki = 510 nM T16016 CDC1Z2 10554359 Ki = 233 nM T16016 CAFS58 10555067 IC50 = 1800 nM T16016 C0CM5H 10555107 IC50 = 2.5 nM T16016 C83NYU 10555351 IC50 = 150 nM T16016 CWS49E 10571296 Ki = 429 nM T16016 COE8I1 10572669 Ki = 98 nM T16016 C6YW1U 10573219 Ki = 463 nM T16016 C0GWC7 10575889 Ki = 78 nM T16016 COM01N 10576419 Ki = 99 nM T16016 C15TUC 10579692 IC50 = 5 nM T16016 CUG16A 10580014 IC50 = 17 nM T16016 C05PCB 10591473 IC50 > 50000 nM T16016 CE1O4F 10596333 Ki = 371 nM T16016 C9J3PF 10597049 Ki = 359 nM T16016 C4KXS5 10599794 Ki = 1155 nM T16016 C53DCW 10623381 Ki = 244 nM T16016 CYE90Z 10643770 Ki = 790 nM T16016 C2DF5Z 10645313 Ki = 206 nM T16016 CJV7U8 10645391 Ki = 1425 nM T16016 CKBR38 10647579 Ki = 330 nM T16016 CRKL63 10649043 Ki = 32 nM T16016 C2CAG8 10652532 IC50 = 3.9 nM T16016 CV27LS 10667913 Ki = 533 nM T16016 CS93VO 10670301 IC50 = 51 nM T16016 CH65OG 10670785 Ki = 347 nM T16016 CND87M 10672205 Ki = 3430 nM T16016 C3BM7V 10676519 IC50 = 3.3 nM T16016 CB4PJ6 10690854 Ki = 236 nM T16016 C4U5IV 10693630 Ki = 7500 nM T16016 CY4D2Q 10694874 Ki = 400 nM T16016 CGL09P 10695227 Ki = 497 nM T16016 C0Q3PC 10695296 IC50 = 800 nM T16016 C80BGV 10698567 IC50 = 2 nM T16016 CT02HZ 10717972 Ki = 33 nM T16016 CAYG15 10722082 Ki = 8 nM T16016 COMN02 10737864 Ki = 584 nM T16016 C60FAV 10741203 IC50 > 10000 nM T16016 CK2VW3 10742114 IC50 > 10000 nM T16016 C5CPM3 10743274 Ki = 153 nM T16016 CNX07L 10764931 Ki = 53 nM T16016 C7I2NG 10765199 IC50 = 140 nM T16016 C3XVO7 10766333 Ki = 234 nM T16016 C68ILN 10766998 Ki = 74 nM T16016 CFV5B7 10767747 IC50 > 10000 nM T16016 C3P9OQ 10768343 Ki = 623 nM T16016 C02OLI 10769446 IC50 = 14 nM T16016 CS2JC3 10786180 Ki = 460 nM T16016 CBMA67 10788075 Ki = 1020 nM T16016 C6G7KV 10789018 Ki = 92 nM T16016 CXVY80 10789482 Ki = 51 nM T16016 C5QU0S 10793529 IC50 = 5100 nM T16016 C6XEU2 10809142 Ki = 1000 nM T16016 CTB07E 10810107 Ki = 975 nM T16016 C9AST2 10811393 Ki = 125 nM T16016 CG8FW4 10811980 IC50 = 1100 nM T16016 C6DCL5 10812461 Ki = 136 nM T16016 CSN93A 10813846 Ki = 715 nM T16016 CZX0G4 10814504 Ki = 406 nM T16016 CN0W4S 10816698 IC50 = 800 nM T16016 CRZ43V 10833944 Ki = 156 nM T16016 CE0JO2 10837160 Ki = 366 nM T16016 C36WKP 10838033 Ki = 405 nM T16016 C9EZ4N 10873705 IC50 = 260 nM T16016 C47TRP 10875472 IC50 = 167 nM T16016 C6HE2M 10916572 IC50 > 50000 nM T16016 C0EM4G 10928173 IC50 > 10000 nM T16016 CX1GK6 10928228 IC50 > 50000 nM T16016 C86DMO 10934382 IC50 > 50000 nM T16016 CX2K8E 10974378 IC50 = 310 nM T16016 CB2CG7 10984360 IC50 > 10000 nM T16016 CN87LP 10985078 IC50 = 890 nM T16016 CZM5K3 10993686 IC50 > 10000 nM T16016 CWS9J7 10995218 IC50 = 31 nM T16016 CDO30J 10995329 IC50 = 240 nM T16016 CPC19I 11004663 IC50 > 10000 nM T16016 CGY15F 11015975 IC50 > 10000 nM T16016 CK70OY 11026367 IC50 > 10000 nM T16016 C82RPC 11026461 IC50 > 50000 nM T16016 CJGS81 11026634 IC50 > 10000 nM T16016 CNE74S 11037958 IC50 = 450 nM T16016 CZ3CB6 11048445 IC50 > 10000 nM T16016 C9UK2E 11049424 IC50 < 780 nM T16016 CVX0M9 11060510 IC50 < 780 nM T16016 C8JG0H 11060814 IC50 < 780 nM T16016 CL82DR 11069916 IC50 > 10000 nM T16016 CH0DL9 11072063 IC50 = 780 nM T16016 CSUH61 11072275 IC50 = 500 nM T16016 CFG06R 11082578 IC50 = 1340 nM T16016 CCD3L5 11091447 IC50 > 10000 nM T16016 C90YHK 11104005 IC50 = 360 nM T16016 C4FB5K 11113940 IC50 = 3600 nM T16016 CZ9U7O 11124782 IC50 = 125 nM T16016 C9P3ME 11133428 IC50 > 10000 nM T16016 CIP20Q 11134412 IC50 > 10000 nM T16016 CWJ69P 11166434 IC50 = 59 nM T16016 C8L4JY 11211557 IC50 = 600 nM T16016 CA39QR 11227406 IC50 > 10000 nM T16016 CW6S9U 11236656 IC50 = 50 nM T16016 CQ6KW0 11272103 IC50 = 10000 nM T16016 C06TUD 11285791 IC50 > 10000 nM T16016 C1A5ET 11329244 IC50 = 10000 nM T16016 C8I2LV 11351191 IC50 = 16 nM T16016 C2L8BH 11397004 IC50 = 6 nM T16016 C39QNY 11464915 IC50 = 32 nM T16016 CY7S2M 11554849 IC50 = 10 nM T16016 C1HAT5 11719164 IC50 = 200 nM T16016 C3KU0D 11722772 IC50 > 50000 nM T16016 CB34MH 11729258 IC50 > 50000 nM T16016 CVB47P 11733139 IC50 > 10000 nM T16016 CVLM30 11734303 IC50 = 71 nM T16016 CPG15O 11743399 IC50 = 1 nM T16016 CL54BJ 11744314 IC50 = 0.36 nM T16016 CQN35J 11764610 IC50 = 7.9 nM T16016 CI29EG 11794863 IC50 = 510 nM T16016 CU1EP6 11798220 Ki = 908 nM T16016 CTB87F 11801019 Ki = 6 nM T16016 C0B9XN 11803141 IC50 = 1.9 nM T16016 CSX85G 11811443 IC50 > 10000 nM T16016 COZ69K 11813735 IC50 = 67 nM T16016 CT8D3H 11814253 IC50 = 1410 nM T16016 CO23LC 11825113 IC50 > 10000 nM T16016 C96ZJD 11828013 IC50 < 780 nM T16016 C6QN3V 11828215 IC50 = 295 nM T16016 C5F3ZC 12015739 IC50 = 11800 nM T16016 C8BM0H 12041800 EC50 = 2000 nM T16016 CRY83B 12093162 Ki = 251.19 nM T16016 C2QWR3 12093163 Ki = 489.78 nM T16016 C79CBJ 12093167 Ki = 15 nM T16016 C3E1FW 12112109 IC50 = 8 nM T16016 CK80NA 12987698 EC50 = 4900 nM T16016 CJGC50 14434082 IC50 < 1000000 nM T16016 CV3O8X 14770534 IC50 > 32000 nM T16016 C7X3CQ 15604497 Ki = 1000 nM T16016 CIZ8C1 15783796 EC50 = 1258.93 nM T16016 CQJ7Y2 15985912 Ki = 398.11 nM T16016 C0G1SC 15985914 Ki = 501.19 nM T16016 C8IKY6 17553211 IC50 > 3000 nM T16016 C9EHC5 17753030 IC50 = 7 nM T16016 CRM90U 19430534 Ki = 501.19 nM T16016 C1ZYS2 21070982 IC50 = 182 nM T16016 C13PWC 21070983 IC50 = 12 nM T16016 C0AOI7 21070984 IC50 = 77 nM T16016 C1CA6D 21070989 IC50 = 2.5 nM T16016 C7FA0C 21070990 IC50 = 3400 nM T16016 CB03CZ 21070993 IC50 = 100 nM T16016 CM27EA 21071046 IC50 = 340 nM T16016 CU8Q7B 21071066 IC50 = 5600 nM T16016 C28JBU 21071070 IC50 = 1100 nM T16016 CV6NF4 21071081 IC50 = 11000 nM T16016 CNM1A8 21071083 IC50 = 2700 nM T16016 C2AS6B 21071094 IC50 = 98 nM T16016 C4WI1R 21071096 IC50 = 32000 nM T16016 C57SVE 21071098 IC50 = 5650 nM T16016 CWMA26 21071099 IC50 = 9800 nM T16016 CZT7J5 21071106 IC50 = 3300 nM T16016 CVQU01 21071108 IC50 = 3650 nM T16016 CC9YA1 22335665 Ki = 47.86 nM T16016 CTO2A8 22335694 Ki = 42.66 nM T16016 CKO01W 22725647 Ki = 30.9 nM T16016 CRM12J 23283073 IC50 = 9.7 nM T16016 C27VNB 24712289 IC50 > 3000 nM T16016 C0J1HA 24738063 IC50 = 4.1 nM T16016 C48OHP 24740167 IC50 = 525 nM T16016 CYX72D 24740170 IC50 = 375 nM T16016 C25HKJ 24758044 IC50 = 28 nM T16016 CW2CM4 24758045 IC50 = 26 nM T16016 C8KC5X 24758046 IC50 = 118 nM T16016 CJF53V 24758047 IC50 = 70 nM T16016 CC7N3T 24758171 IC50 = 40 nM T16016 C1JHY4 24758172 IC50 = 32 nM T16016 C8F0CE 24758173 IC50 = 32 nM T16016 C0P3BR 24758174 IC50 = 24 nM T16016 CXE3M1 24758175 IC50 = 58 nM T16016 C2EP9Y 24758176 IC50 = 25 nM T16016 CA5C3R 24758294 IC50 = 30 nM T16016 C7UE5H 24758295 IC50 = 8 nM T16016 C0OU9Z 24758296 IC50 = 13 nM T16016 CD0XB9 24758297 IC50 = 14 nM T16016 CQ9WX7 24758298 IC50 = 18 nM T16016 CI0V6U 24758299 IC50 = 19 nM T16016 CKH7M2 24758406 IC50 = 20 nM T16016 C93QGZ 24758408 IC50 = 22 nM T16016 CIY5Q4 24758517 IC50 = 44 nM T16016 C32AZH 24758518 IC50 = 45 nM T16016 CD5JH7 24758630 IC50 = 121 nM T16016 CS6NW4 24758743 IC50 = 152 nM T16016 C7ZRE8 24758744 IC50 = 50 nM T16016 C6F1NH 24758745 IC50 = 85 nM T16016 CF9S7E 24758856 IC50 = 40 nM T16016 C9H6MY 24759081 IC50 = 35 nM T16016 C5YDC2 24759191 IC50 = 36 nM T16016 CF6GO2 24759420 IC50 = 80 nM T16016 C6CET2 24759740 IC50 = 388 nM T16016 CPD05R 24782574 IC50 = 50 nM T16016 CISV81 24782826 IC50 = 22 nM T16016 CLG7M5 25022507 IC50 = 90 nM T16016 C7NJ1B 25109291 Ki = 0.043 nM T16016 C54LQF 25230828 IC50 > 50000 nM T16016 CZX9B0 25231298 IC50 > 75000 nM T16016 C74EOA 25231299 IC50 = 3600 nM T16016 C98VPY 25231300 IC50 = 270 nM T16016 CF76KB 25231301 IC50 = 270 nM T16016 CZXC46 25231302 IC50 = 43000 nM T16016 C0RZJ5 25231303 IC50 > 100000 nM T16016 C2J4GS 25231477 IC50 > 13000 nM T16016 C6YW9F 25231478 IC50 > 77000 nM T16016 C6JNK1 25231479 IC50 > 100000 nM T16016 CRP1H8 25231480 IC50 = 1300 nM T16016 C9H2LY 25231481 IC50 = 5700 nM T16016 COHI45 25231482 IC50 > 100000 nM T16016 C5C8DA 25233577 IC50 = 4000 nM T16016 CIX06B 25233578 IC50 = 4700 nM T16016 CVCF50 25233579 IC50 = 680 nM T16016 CE1FK6 25233580 IC50 = 700 nM T16016 CD8F7W 25233581 IC50 = 720 nM T16016 CEF52O 25233582 IC50 = 290 nM T16016 C8H5EP 25233753 IC50 = 2950 nM T16016 CAL67P 25233754 IC50 = 120 nM T16016 CNVF07 25233755 IC50 = 22 nM T16016 C8W5VE 25233756 IC50 = 6 nM T16016 CCGL97 25233757 IC50 > 28000 nM T16016 C72FBZ 25233758 IC50 > 100000 nM T16016 C3CAP1 25233941 IC50 > 28000 nM T16016 CDJ67K 25233947 IC50 = 540 nM T16016 C07BSM 25252974 IC50 = 4 nM T16016 CS0XW4 25253284 IC50 = 20 nM T16016 CUKC71 25254218 IC50 = 22 nM T16016 C8E3GU 26042546 IC50 > 30000 nM T16016 CQD8U5 31900420 IC50 > 3000 nM T16016 CIKC26 32637491 IC50 > 3000 nM T16016 C5D0XT 36715516 IC50 > 3000 nM T16016 CXI89R 37664972 IC50 = 790 nM T16016 CC3D2Q 40636824 IC50 > 3000 nM T16016 CA79PZ 40636827 IC50 > 3000 nM T16016 CAR7X3 42602328 IC50 = 1.8 nM T16016 C8A5TC 42602331 IC50 = 1.4 nM T16016 CU2PO5 44180522 IC50 > 25118.86 nM T16016 C5YFB9 44252324 IC50 > 10000 nM T16016 CKNR65 44281427 IC50 = 370 nM T16016 CPS75A 44308794 IC50 < 50000 nM T16016 C0MU9T 44308812 IC50 < 50000 nM T16016 CJZ54H 44308819 IC50 = 840 nM T16016 C1T9VK 44308837 IC50 < 50000 nM T16016 CW29KX 44308850 IC50 < 50000 nM T16016 C03USP 44308902 IC50 = 30000 nM T16016 C2MA1N 44308997 IC50 = 2490 nM T16016 CCRW52 44309046 IC50 > 32000 nM T16016 CBC5G2 44309060 IC50 = 10300 nM T16016 CI4P5Z 44309061 IC50 = 55100 nM T16016 CW2JL5 44309067 IC50 < 50000 nM T16016 CDF92Y 44309074 IC50 = 64 nM T16016 C8O0UX 44309077 IC50 = 5600 nM T16016 CWXN65 44309087 IC50 = 18500 nM T16016 C9K2EI 44309091 IC50 = 8000 nM T16016 CWNB28 44309094 IC50 > 32000 nM T16016 CJ3WS4 44309105 IC50 = 280 nM T16016 CW3FI1 44309112 IC50 = 5150 nM T16016 COK2M0 44309119 IC50 < 50000 nM T16016 CF28NB 44309120 IC50 > 32000 nM T16016 CPTJ37 44309122 IC50 = 27 nM T16016 C3NG7S 44309124 IC50 = 740 nM T16016 C49FZD 44309128 IC50 = 4600 nM T16016 COWL46 44309136 IC50 < 50000 nM T16016 CC5ZE8 44309143 IC50 = 1 nM T16016 C81JTN 44309155 IC50 = 15000 nM T16016 C41TRZ 44309156 IC50 < 50000 nM T16016 CE52DG 44309161 IC50 = 3460 nM T16016 C7UV9B 44309163 IC50 = 22 nM T16016 CYE9C4 44309165 IC50 = 15 nM T16016 C3ZD4J 44309166 IC50 = 3500 nM T16016 CVA24D 44309171 IC50 = 420 nM T16016 C0XA4Q 44309178 IC50 = 2600 nM T16016 CJSP94 44309185 IC50 = 670 nM T16016 C3SHY2 44309192 IC50 = 610 nM T16016 C93LQN 44309194 IC50 = 580 nM T16016 C2ENG9 44309195 IC50 = 20 nM T16016 CRU6E3 44309213 IC50 = 2900 nM T16016 C2P1KQ 44309219 IC50 = 560 nM T16016 CT7DV5 44309222 IC50 = 4200 nM T16016 C7KLP0 44309235 IC50 = 580 nM T16016 CL8P6W 44309236 IC50 = 510 nM T16016 C6V8DR 44309237 IC50 = 16700 nM T16016 CVIJ87 44309244 IC50 = 44800 nM T16016 CU52KE 44309245 IC50 = 850 nM T16016 C0GY2J 44309267 IC50 = 130 nM T16016 CE2I6H 44309286 IC50 = 7 nM T16016 C71LNC 44309312 IC50 = 8 nM T16016 CGDF80 44309313 IC50 = 52 nM T16016 CA5YD0 44309318 IC50 = 48 nM T16016 CHS3F9 44309327 IC50 = 26 nM T16016 C8CY4Z 44309337 IC50 = 8 nM T16016 CXQ38W 44309347 IC50 = 160 nM T16016 C7B5LR 44309353 IC50 = 46 nM T16016 CVO98N 44309364 IC50 = 130 nM T16016 C8DTH6 44309365 IC50 > 25000 nM T16016 CPQ8T7 44309397 IC50 = 9 nM T16016 C27LRK 44309407 IC50 = 540 nM T16016 CNQ0G4 44309414 IC50 = 2570 nM T16016 CJFV61 44361881 Ki = 29 nM T16016 CR5S9Y 44362079 Ki = 1188 nM T16016 C8C9LX 44405180 IC50 = 360 nM T16016 C8TS2N 44405181 IC50 = 2.4 nM T16016 CO16BT 44405194 IC50 = 1700 nM T16016 C47JTD 44405196 IC50 = 800 nM T16016 C87DSA 44405202 IC50 = 9.6 nM T16016 CGKV93 44405203 IC50 = 28 nM T16016 C4FS7U 44405211 IC50 = 300 nM T16016 CLDC78 44405212 IC50 = 6 nM T16016 CP3O7Y 44405234 IC50 = 1600 nM T16016 C9ZT8S 44430713 IC50 = 18 nM T16016 CM1E0I 44430714 IC50 = 350 nM T16016 CPI3C7 44430715 IC50 = 78 nM T16016 C53WIQ 44430716 IC50 = 270 nM T16016 CNAZ59 44430717 IC50 = 97 nM T16016 CMJ8I2 44430718 IC50 = 2340 nM T16016 CNA21M 44430720 IC50 = 2910 nM T16016 CKA2R9 44430721 IC50 = 200 nM T16016 C61NLQ 44430722 IC50 = 920 nM T16016 CG9E5H 44430723 IC50 = 14 nM T16016 CQKT60 44430724 IC50 = 160 nM T16016 CBVJ95 44430725 IC50 = 90 nM T16016 CG49JY 44430726 IC50 = 140 nM T16016 CE5AF1 44430727 IC50 > 10000 nM T16016 CSG7K4 44430732 IC50 = 72 nM T16016 CZ9WM3 44430735 IC50 = 170 nM T16016 CWLX40 44430736 IC50 = 800 nM T16016 CV62CF 44430742 IC50 = 160 nM T16016 C8PK5W 44430745 IC50 = 54 nM T16016 CC6YP2 44430746 IC50 = 13 nM T16016 CPM05Z 44430748 IC50 = 6 nM T16016 C9BE1D 44430750 IC50 = 64 nM T16016 CU39TN 44430752 IC50 = 12 nM T16016 CP37VK 44430753 IC50 = 5 nM T16016 C47MRZ 44430754 IC50 = 15 nM T16016 CQSY30 44430755 IC50 = 8 nM T16016 C9BVX3 44430756 IC50 = 26 nM T16016 CSH43L 44430758 IC50 = 6 nM T16016 CF4EM2 44430759 IC50 = 76 nM T16016 CX2Q8V 44430836 IC50 = 220 nM T16016 CQGX84 44431523 IC50 = 480 nM T16016 CU9V8X 44431524 IC50 = 30 nM T16016 C4VN5J 44431527 IC50 = 38 nM T16016 CU42MW 44431528 IC50 = 44 nM T16016 CNZ4R0 44431529 IC50 = 13 nM T16016 C68QOX 44453084 IC50 = 1650 nM T16016 C4QAH9 44453157 IC50 = 390 nM T16016 C5URL9 44453161 IC50 = 280 nM T16016 CZ6QR5 44453162 IC50 = 120 nM T16016 CH9D7P 44453163 IC50 = 7330 nM T16016 CYN36R 44453164 IC50 = 190 nM T16016 C62OVR 44453165 IC50 = 3650 nM T16016 C6HVU9 44453167 IC50 = 2200 nM T16016 CEY32C 44453195 IC50 = 2260 nM T16016 C3VK9H 44453197 IC50 = 2260 nM T16016 CA70QE 44453198 IC50 = 4650 nM T16016 C1QZE2 44453199 IC50 = 120 nM T16016 CAO60C 44453200 IC50 = 50 nM T16016 CXZ96H 44453202 IC50 = 30 nM T16016 CL2YO8 44453225 IC50 = 970 nM T16016 CZ85CL 44453226 IC50 = 670 nM T16016 C1RMH2 44453227 IC50 = 330 nM T16016 CW82CO 44453228 IC50 = 80 nM T16016 CHW4U3 44453229 IC50 = 210 nM T16016 C8NX4K 44453263 IC50 = 370 nM T16016 CSA8W9 44453265 IC50 = 380 nM T16016 CT5LK7 44453289 IC50 > 10000 nM T16016 CRP5D2 44453290 IC50 = 370 nM T16016 CUE83S 44453291 IC50 = 110 nM T16016 CHSC39 44453292 IC50 = 180 nM T16016 CASM45 44453293 IC50 = 140 nM T16016 CMVW23 44453317 IC50 = 7980 nM T16016 CE3UW0 44453320 IC50 = 200 nM T16016 CYA2S8 44453321 IC50 = 420 nM T16016 CJL5T4 44453356 IC50 > 10000 nM T16016 CRM58W 44453357 IC50 = 1240 nM T16016 C4DY0R 44453359 IC50 = 90 nM T16016 C59PBZ 44453361 IC50 = 40 nM T16016 C1VA0H 44453363 IC50 = 180 nM T16016 CQPG50 44453399 IC50 > 10000 nM T16016 CE1PR7 44453400 IC50 = 100 nM T16016 CJIZ23 44453401 IC50 > 10000 nM T16016 CZY72M 44453402 IC50 = 1340 nM T16016 CRN83S 44453403 IC50 = 30 nM T16016 CX4PU5 44453433 IC50 = 1850 nM T16016 CT3D4B 44453435 IC50 = 280 nM T16016 CI9BZ7 44453436 IC50 = 520 nM T16016 CT9D0R 44453437 IC50 = 360 nM T16016 CV0KP8 44453464 IC50 = 1330 nM T16016 C35SCE 44453466 IC50 = 430 nM T16016 C8I5SN 44453467 IC50 = 180 nM T16016 C15TOP 44453469 IC50 = 510 nM T16016 CKX1I6 44453472 IC50 > 1000 nM T16016 C58PQU 44453499 IC50 = 510 nM T16016 CK9E6M 44453501 IC50 = 180 nM T16016 CC7XV8 44453502 IC50 = 6210 nM T16016 CX12CN 44453503 IC50 = 350 nM T16016 C2OED7 44453504 IC50 = 240 nM T16016 CO4ZW0 44453525 IC50 = 1170 nM T16016 CD4Y8C 44453527 IC50 = 1000 nM T16016 CO8TK2 44453528 IC50 = 385 nM T16016 C6G3XF 44453529 IC50 = 160 nM T16016 C1V0EH 44453557 IC50 = 600 nM T16016 CI9E5K 44453559 IC50 > 30000 nM T16016 CDHV21 44453579 IC50 = 400 nM T16016 CV6TD4 44453584 IC50 = 84 nM T16016 C4SLA8 44453611 IC50 > 30000 nM T16016 CMCN57 44453612 IC50 > 10000 nM T16016 C4EM8C 44453614 IC50 = 1400 nM T16016 CUP6R8 44453615 IC50 = 1300 nM T16016 C7CMI0 44453637 IC50 = 1900 nM T16016 CD5QK4 44453638 IC50 = 1290 nM T16016 C2Z1YR 44453639 IC50 = 480 nM T16016 CBA20D 44453641 IC50 = 3880 nM T16016 CL2WB7 44468439 IC50 > 3000 nM T16016 C94VWK 44468440 IC50 = 1200 nM T16016 C5OIK9 44468442 IC50 = 1200 nM T16016 CYXR38 44468570 IC50 = 68 nM T16016 CX6U4M 44468708 IC50 = 61 nM T16016 CR6W8U 44469380 IC50 = 2500 nM T16016 C4DL5C 44469677 IC50 > 10000 nM T16016 CO3D8M 44469804 IC50 = 120 nM T16016 C35AHO 44469942 IC50 = 44 nM T16016 CHE1A2 44470083 IC50 = 5 nM T16016 CHNM79 44470374 IC50 = 12 nM T16016 CA7V8M 44480348 IC50 = 47 nM T16016 C3UMK5 44480600 IC50 = 15 nM T16016 CT5N4E 44555481 IC50 > 50000 nM T16016 CS9U6X 44560288 IC50 = 9.6 nM T16016 CF5X2U 45138007 IC50 = 3 nM T16016 CK50UD 45138010 IC50 = 34 nM T16016 CID15S 45138012 IC50 = 450 nM T16016 C6A3XH 45138458 IC50 = 19 nM T16016 CXC4M1 45138759 IC50 = 0.3 nM T16016 CK3N1G 46206137 IC50 > 10000 nM T16016 CQ3FX0 46858281 IC50 = 2400 nM T16016 C80WVI 49796696 Ki = 206 nM T16016 CVY1G2 49796697 Ki = 116 nM T16016 C95CPY 49798264 Ki = 316.23 nM T16016 C3SUN1 49798265 Ki = 125.89 nM T16016 CBG4T2 49798289 Ki = 125.89 nM T16016 C6C8AV 49865900 IC50 = 16 nM T16016 C87BYU 49865901 IC50 = 810 nM T16016 CJV7Z9 49865951 IC50 = 2.9 nM T16016 C8K6CQ 52916803 IC50 = 1.8 nM T16016 C3P7QF 52917500 IC50 = 2 nM T16016 C0NT2M 52932654 IC50 > 3000 nM T16016 CCI58B 54712652 Ki = 199.53 nM T16016 CH3UL5 57390926 IC50 = 261 nM T16016 CK2Y8P 57396208 IC50 = 387 nM T16016 CR09LY 57400127 IC50 > 25118.86 nM T16016 CAT9F4 57840192 IC50 = 10 nM T16016 CT1JC7 57840210 IC50 = 5200 nM T16016 CTAH32 57840282 IC50 = 20 nM T16016 CJ90DZ 57840295 IC50 = 10 nM T16016 C4RC3N 57840302 IC50 = 6 nM T16016 C3LMG6 57840312 IC50 = 120 nM T16016 C9QO4L 57840315 IC50 = 97 nM T16016 C89RVZ 57840356 IC50 = 18 nM T16016 C5S7FB 57840363 IC50 = 2 nM T16016 CVW80D 57840380 IC50 = 68 nM T16016 CFJ80G 57840427 IC50 = 40 nM T16016 CE3V0N 57840435 IC50 = 8 nM T16016 C9KW6F 57840437 IC50 = 5 nM T16016 CNA3W0 57840460 IC50 = 92 nM T16016 CFS8P5 57840482 IC50 = 7 nM T16016 CM6UK5 57840511 IC50 = 10 nM T16016 C5CU2J 57840512 IC50 = 23 nM T16016 CM32AV 57840515 IC50 = 47 nM T16016 CD5Z6H 57840518 IC50 = 37 nM T16016 C4I2OZ 57840522 IC50 = 740 nM T16016 CI2B1E 57840556 IC50 = 19 nM T16016 CI6XW0 57840557 IC50 = 500 nM T16016 C25SLU 57888652 IC50 = 130 nM T16016 C7TBL8 57888663 IC50 = 233 nM T16016 CM31AW 57888688 IC50 = 303 nM T16016 C6NLY7 57888690 IC50 = 46 nM T16016 CTX8J4 57888707 IC50 = 107 nM T16016 CTY08U 57888715 IC50 = 100 nM T16016 C1EGP2 57888718 IC50 = 1077 nM T16016 CD08VL 57888746 IC50 = 194 nM T16016 CUX61B 57888747 IC50 = 4.7 nM T16016 C70ZKN 57888758 IC50 = 2940 nM T16016 C32IGS 57888775 IC50 = 152 nM T16016 CUG73D 57888785 IC50 = 6 nM T16016 CD8XO3 57888812 IC50 = 259 nM T16016 CQ79WS 57888832 IC50 = 115 nM T16016 CBS39N 57888834 IC50 = 1.7 nM T16016 CG15IU 57888886 IC50 = 854 nM T16016 CGK3S6 57888895 IC50 = 3.3 nM T16016 C7USZ8 57888900 IC50 = 9.9 nM T16016 CSR0N6 57888907 IC50 = 2 nM T16016 C7S5XP 57888919 IC50 = 0.8 nM T16016 CG3JO6 57888925 IC50 = 262 nM T16016 C14OID 57888938 IC50 = 40 nM T16016 CWKP07 57888949 IC50 = 616 nM T16016 CUHR07 57888953 IC50 = 55 nM T16016 C8EBZ4 57888963 IC50 = 370 nM T16016 C56BOX 57888966 IC50 = 9.9 nM T16016 C9FM2N 57888993 IC50 = 1 nM T16016 C05HEB 57889002 IC50 = 423 nM T16016 COP15F 57889003 IC50 = 0.8 nM T16016 CO67FJ 57889006 IC50 = 539 nM T16016 CUCX67 57889023 IC50 = 3.4 nM T16016 C4VC6R 57889047 IC50 = 20 nM T16016 CCD01J 57889071 IC50 = 1.8 nM T16016 CLT76V 57889077 IC50 = 2.2 nM T16016 CCQ8G1 57889099 IC50 = 2 nM T16016 C69CJK 57889121 IC50 = 4.4 nM T16016 CW4S5A 57889141 IC50 = 180 nM T16016 CBMJ90 57889158 IC50 = 15 nM T16016 CM8IY2 57889164 IC50 = 2.9 nM T16016 CP13VI 57889180 IC50 = 4 nM T16016 CMZQ02 57889181 IC50 = 3 nM T16016 C1J5RH 57889188 IC50 = 3 nM T16016 CH9V4I 57889230 IC50 = 1.7 nM T16016 CY9F3C 57889234 IC50 = 933 nM T16016 CUW9Z5 57889255 IC50 = 140 nM T16016 CPD8S4 57889291 IC50 = 7.6 nM T16016 CJ5C3D 57889314 IC50 = 3 nM T16016 CMT6C1 57889327 IC50 = 1 nM T16016 CDOA16 57889334 IC50 = 1.9 nM T16016 C4DMF2 57889346 IC50 = 543 nM T16016 C9SR2K 57889347 IC50 = 2.6 nM T16016 C9AMN1 57889407 IC50 = 341 nM T16016 CN0WX5 57889423 IC50 = 2.5 nM T16016 C0YCH2 57889430 IC50 = 1.1 nM T16016 C5EU1V 57889478 IC50 = 45 nM T16016 CM9PI7 57889484 IC50 = 153 nM T16016 CFOK45 57889591 IC50 = 120 nM T16016 C8KEZ3 57889592 IC50 = 185 nM T16016 C26KEZ 57889613 IC50 = 10 nM T16016 CF2E5A 57889625 IC50 = 191 nM T16016 CJ2P3S 57889635 IC50 = 9 nM T16016 CY28OV 57889649 IC50 = 7.1 nM T16016 C0AOP9 57889660 IC50 = 13 nM T16016 C70YGB 57889664 IC50 = 105 nM T16016 C7OQV8 57889667 IC50 = 172 nM T16016 CW4Q2Z 57889679 IC50 = 10 nM T16016 C5G6PM 57889696 IC50 = 121 nM T16016 C31ZKO 57889736 IC50 = 3 nM T16016 CL29GA 57889758 IC50 = 5.8 nM T16016 CA46BV 57889764 IC50 = 1.2 nM T16016 CL8GT3 57889796 IC50 = 180 nM T16016 CLKA82 57889843 IC50 = 3.6 nM T16016 C7ZF9O 57889874 IC50 = 265 nM T16016 C3SZL5 57889880 IC50 = 521 nM T16016 CNV92I 57889883 IC50 = 70 nM T16016 CX82KS 57889897 IC50 = 4.1 nM T16016 C7KL5M 57889944 IC50 = 88 nM T16016 C9U8JV 57889972 IC50 = 324 nM T16016 C4Z3GA 57889974 IC50 = 6.3 nM T16016 CG1M7U 57889975 IC50 = 18 nM T16016 C9LKQ5 57889979 IC50 = 4.3 nM T16016 C9VE5T 57991685 IC50 = 1603 nM T16016 CAL9F2 57991690 IC50 = 95 nM T16016 CLH4Y8 57991707 IC50 = 2.3 nM T16016 CUNM10 57991713 IC50 = 208 nM T16016 CBQ7I3 58138764 IC50 > 3000 nM T16016 C84IXN 58138765 IC50 = 1100 nM T16016 CPWO40 58138766 IC50 > 3000 nM T16016 CIP73G 58138781 IC50 = 450 nM T16016 CY5G6S 58138788 IC50 = 750 nM T16016 C7IVB1 58138789 IC50 = 4.5 nM T16016 C1PAV2 58138800 IC50 > 3000 nM T16016 C1FV4A 58138826 IC50 = 22 nM T16016 CW20DR 58138832 IC50 = 1700 nM T16016 CM3L2A 58138839 IC50 > 3000 nM T16016 CQXC68 58138841 IC50 = 55 nM T16016 CKMW80 58138845 IC50 = 210 nM T16016 C6I3ED 58138852 IC50 = 170 nM T16016 C12JLA 58138868 IC50 = 17 nM T16016 CFHQ71 58138880 IC50 = 6 nM T16016 CNG5X3 58138893 IC50 = 180 nM T16016 CD01TW 58138911 IC50 = 260 nM T16016 C0YWT1 58509213 IC50 > 10000 nM T16016 C5P0GD 58778003 IC50 = 8 nM T16016 C08OME 58778007 IC50 = 6400 nM T16016 C0I2HN 59278115 IC50 = 1.4 nM T16016 CJW8D2 59278123 IC50 = 8 nM T16016 C8CZ7T 59278147 IC50 = 1.2 nM T16016 C03SHK 59278235 IC50 = 61 nM T16016 C4KU2S 59278286 IC50 = 0.2 nM T16016 CRH6S5 59278305 IC50 = 12 nM T16016 CA23BD 59278307 IC50 = 12 nM T16016 CEAY32 59278314 IC50 = 6.8 nM T16016 C1L2SC 59278332 IC50 = 0.2 nM T16016 CLS59N 59278436 IC50 = 2 nM T16016 CO78WQ 59278474 IC50 = 41 nM T16016 CK2CB9 59687824 IC50 = 5 nM T16016 CODB07 66686405 IC50 = 0.8 nM T16016 CO74RQ 68416145 IC50 > 3000 nM T16016 CG46AF 68816399 IC50 = 560 nM T16016 CQ34PJ 68817337 IC50 = 32 nM T16016 CAN47O 68818375 IC50 = 9 nM T16016 C9S1NP 68818964 IC50 = 79 nM T16016 C6KH1J 68956901 IC50 = 7.1 nM T16016 CRWB79 68958915 IC50 = 130 nM T16016 CZHF19 68959770 IC50 = 1.4 nM T16016 C8HM7E 68959963 IC50 = 0.36 nM T16016 C3H9CD 68962095 IC50 = 5 nM T16016 C8Y3PB 68963393 IC50 = 2.5 nM T16016 C1E4QF 68963562 IC50 = 12 nM T16016 C1KAN5 68963686 IC50 = 1.1 nM T16016 C52BVJ 68963698 IC50 = 89 nM T16016 C6Z7UL 69435853 IC50 = 7.1 nM T16016 CQVW46 69437029 IC50 = 160 nM T16016 CNY8G5 69437067 IC50 = 1300 nM T16016 C37WGU 69437285 IC50 = 560 nM T16016 C6XQ3C 69439557 IC50 = 37 nM T16016 CG3DM1 71214709 Ki = 398.11 nM T16016 CG5V6I 71214710 Ki = 1584.89 nM T16016 CA72CU 71214725 Ki = 1000 nM T16016 CMSH09 71214976 Ki = 1258.93 nM T16016 CSD6R9 71450657 Ki = 501.19 nM T16016 C8A0XW 71450658 Ki = 316.23 nM T16016 C4SH7L 71452035 IC50 = 177 nM T16016 C8YW2L 71452487 Ki = 1584.89 nM T16016 C1TOE8 71452488 Ki = 1000 nM T16016 CT7FK3 71453837 IC50 = 66 nM T16016 C71FXH 71454246 Ki = 3981.07 nM T16016 CD8I7C 71454247 Ki = 1584.89 nM T16016 CSL01M 71454248 Ki = 316.23 nM T16016 CSN6K4 71455572 IC50 = 14930 nM T16016 C3EYK5 71456007 Ki = 7943.28 nM T16016 CHV16Z 71456008 Ki = 1584.89 nM T16016 C7K2XU 71457361 IC50 = 38 nM T16016 CCYR75 71457362 IC50 = 34 nM T16016 C6MHX5 71457815 Ki = 2511.89 nM T16016 C76AQC 71460999 IC50 = 2832 nM T16016 C3BXS9 71461438 Ki = 1000 nM T16016 CRV73F 71461439 Ki = 1000 nM T16016 C3P5HM 71461440 Ki = 1000 nM T16016 CIP7D8 71462570 Ki = 2.3 nM T16016 C5E1FJ 71463165 Ki = 7943.28 nM T16016 C8VX0L 71463166 Ki = 1995.26 nM T16016 CTZ63Y 71560163 IC50 = 120 nM T16016 CVH9S8 71570633 IC50 = 0.79 nM T16016 C6ZBW8 71570634 IC50 = 18 nM T16016 C46RFP 71655299 IC50 = 1.3 nM T16016 CUI4D7 71655559 IC50 = 110 nM T16016 CHZ92K 71680936 IC50 = 2.3 nM T16016 CS1X3B 71681244 IC50 = 20 nM T16016 C86DGB 71681399 IC50 = 2.2 nM T16016 CGFZ24 71681400 IC50 = 17 nM T16016 C1IX0A 71682816 IC50 = 2240 nM T16016 CNE87P 71717436 IC50 = 5 nM T16016 CVM47W 71717437 IC50 = 420 nM T16016 C30LKZ 71718022 IC50 = 12 nM T16016 CG18BJ 71718023 IC50 = 16 nM T16016 C5N7RO 71718646 IC50 = 107 nM T16016 CM45XP 71718647 IC50 = 220 nM T16016 CSF0T9 71719253 IC50 = 11 nM T16016 C3EUY7 71719254 IC50 = 14 nM T16016 C9F0XG 71719255 IC50 = 210 nM T16016 C05FBT 71719855 IC50 = 10 nM T16016 CEPD62 71719856 IC50 = 52 nM T16016 CWH6T3 72548703 IC50 = 0.081 nM T16016 C4S2OT 72945111 IC50 = 13 nM T16016 C7MS4G 72945112 IC50 = 3.2 nM T16016 CV74IH 72945310 IC50 = 4.5 nM T16016 CXOI39 72945311 IC50 = 1.3 nM T16016 C5TS1M 72945313 IC50 = 1.8 nM T16016 CH63BO 72945314 IC50 = 1.8 nM T16016 C2VU8F 72945510 IC50 = 0.89 nM T16016 CAO2L3 72945511 IC50 = 2.2 nM T16016 CQ5MD0 72945512 IC50 = 0.63 nM T16016 C42LID 72947880 IC50 = 1300 nM T16016 CWSX63 73345959 IC50 > 8333 nM T16016 CH0R4L 73347500 IC50 = 196 nM T16016 CBWU87 73349030 IC50 = 1800 nM T16016 C9E6RP 73350585 IC50 = 7.2 nM T16016 C15IOL 73353555 IC50 = 25000 nM T16016 CUA0J7 73353556 IC50 > 8333 nM T16016 CR79ZO 73353557 IC50 > 8333 nM T16016 CJ3L5M 73355055 IC50 = 3.7 nM T16016 C7V1JG 76311396 IC50 = 9100 nM T16016 CH7B9N 76311400 IC50 = 260 nM T16016 CGP1F3 76315009 IC50 = 5700 nM T16016 C5IJN1 76318623 IC50 = 12700 nM T16016 C4TYD3 76322249 IC50 = 10000 nM T16016 C2YJR4 76322269 IC50 = 10000 nM T16016 CR4IO8 76325891 IC50 = 4000 nM T16016 CW12KH 76336764 IC50 = 260 nM T16016 CP3C1F 118714001 IC50 = 2 nM T16016 C3P4VQ 118714034 IC50 = 11 nM T16016 C79CKF 118714035 IC50 = 2 nM T16016 CFB78G 118714036 IC50 = 2 nM T16016 CM5F8Z 118714037 IC50 = 2 nM T16016 C2KET6 118714038 IC50 = 2 nM T16016 C5I8EN 134817249 IC50 > 30000 nM T16016 C4Z3XS 145983516 IC50 > 30000 nM T16016 C9NDM5 145983631 IC50 > 30000 nM T16016 C3ZPR5 145985518 IC50 > 30000 nM T16016 CHTY23 145985766 IC50 > 30000 nM T16016 C54YUG 155511496 IC50 > 3000 nM T16016 C3CJ8L 155511620 IC50 = 10 nM T16016 C7R1SZ 155513751 Ki = 40.74 nM T16016 CM7Y9H 155514261 Ki = 50 nM T16016 C7HW9V 155514720 IC50 > 3000 nM T16016 CW1K9P 155515101 IC50 > 3000 nM T16016 CDI07N 155515240 IC50 > 3000 nM T16016 CT45DJ 155515471 IC50 > 3000 nM T16016 CZ29FQ 155521447 Ki = 5 nM T16016 CNH6D0 155522863 IC50 > 3000 nM T16016 C8Q0SV 155526212 IC50 = 350 nM T16016 CW0R6Z 155526680 Ki = 64.57 nM T16016 C86PTC 155528640 IC50 > 3000 nM T16016 CA6QL2 155529800 IC50 > 3000 nM T16016 CDRM08 155530458 IC50 = 1200 nM T16016 C15NKD 155532102 Ki = 181 nM T16016 C7KI0H 155533083 IC50 > 3000 nM T16016 CTW3H0 155533145 IC50 = 1900 nM T16016 CF6DQ7 155535265 Ki = 18.2 nM T16016 CM5R3Q 155538641 IC50 > 3000 nM T16016 CR0A2Y 155538947 IC50 = 28 nM T16016 CE5SU4 155539148 Ki = 30 nM T16016 C0KX7I 155539505 IC50 > 3000 nM T16016 CSP9L2 155543214 IC50 > 3000 nM T16016 COK7D3 155544726 IC50 = 1700 nM T16016 C4J1ZL 155545804 Ki = 31 nM T16016 C0D3CS 155547454 IC50 > 3000 nM T16016 C62DPU 155548977 Ki = 77 nM T16016 CIU9M4 155549273 IC50 = 960 nM T16016 C8DX4C 155549724 IC50 = 500 nM T16016 C0QHR1 155549943 IC50 > 3000 nM T16016 C80MNA 155553428 Ki = 198 nM T16016 C05PNE 155554350 IC50 > 3000 nM T16016 CHX96A 155556819 IC50 > 3000 nM T16016 C7X6VW 155559153 Ki = 27.54 nM T16016 CDUT06 155561022 Ki = 194.98 nM T16016 CC1JE8 155561040 IC50 = 420 nM T16016 CDS87R 155562877 IC50 = 2100 nM T16016 C2KB9Y 155564974 IC50 = 13 nM T16016 CMZ94A 155565119 IC50 > 3000 nM T16016 CY1BK9 155565496 IC50 > 3000 nM T16016 CT6P7E 155566515 IC50 > 3000 nM T16016 CV8IG3 155568751 IC50 > 3000 nM T16016 CT27HO 155569186 IC50 > 3000 nM T16016 D01JZV 9913085 IC50 = 1900 nM T16016 D05XZF 512282 Ki = 1 nM T16016 D06QRP 5311123 IC50 = 39 nM T16016 D0FF6S 16038374 IC50 > 10000 nM T38200 D0ED7U 60648 IC50 = 917000 nM T38200 D08ESA 198693 IC50 = 333000 nM T38200 D0C9XA 119 IC50 = 1000 nM T38200 CJ9V4G 40598 IC50 > 1000000 nM T38200 CXSD61 155246 IC50 = 43700 nM T38200 CHV0G9 639062 IC50 > 1000000 nM T38200 C97FYX 702501 IC50 > 300000 nM T38200 C8X9TQ 1069892 Ki > 100000 nM T38200 C1A0UL 1502074 IC50 = 2300 nM T38200 C3DR8J 1502075 IC50 = 2511.89 nM T38200 C9EI4M 1530639 IC50 > 1000000 nM T38200 CU23IC 4531494 IC50 = 10000 nM T38200 CG1ZF6 5311322 Ki = 6100 nM T38200 CN2C7Q 6604883 IC50 = 86000 nM T38200 C4A6SU 8181355 IC50 > 500000 nM T38200 CQ64IH 9797818 IC50 = 1990000 nM T38200 C31HNE 9884272 Ki > 100000 nM T38200 CY2IS7 9888224 IC50 = 46000 nM T38200 CI06JL 9982662 IC50 = 198000 nM T38200 CTZ5Q7 9983570 IC50 = 1080000 nM T38200 C75BDY 10031163 IC50 = 212000 nM T38200 CZ4PO2 10050339 IC50 = 6740000 nM T38200 CZQ52G 10052359 IC50 = 169000 nM T38200 CP2WF1 10072112 IC50 = 142000 nM T38200 CG1A4H 10073933 IC50 = 25000 nM T38200 C57RVK 10075407 IC50 = 142000 nM T38200 C4S1CO 10096504 IC50 = 25000 nM T38200 CXJR61 10252950 IC50 = 178000 nM T38200 CC8V4E 10412575 IC50 = 20000 nM T38200 CZ8FQ2 10481573 IC50 = 29000 nM T38200 CU40KP 11743493 IC50 = 91000 nM T38200 CH6GX1 13314232 IC50 > 500000 nM T38200 C03OAI 14810154 IC50 = 8128.31 nM T38200 C6VK4E 17173775 IC50 > 1000000 nM T38200 CE92MX 17174058 IC50 > 1000000 nM T38200 C3OQD7 17250318 IC50 > 500000 nM T38200 CME93B 43345728 IC50 > 1000000 nM T38200 C5JUW9 47058964 IC50 > 1000000 nM T38200 CLIK30 50941729 IC50 > 100000 nM T38200 CQ4XJ7 55285849 IC50 = 13900 nM T38200 CY9O8W 55285850 IC50 = 13900 nM T38200 C8UTR2 67642717 IC50 = 1900 nM T38200 C6ME5H 70684991 IC50 = 876000 nM T38200 C79CYX 70689234 IC50 = 2043000 nM T38200 CD9EV5 70691307 IC50 = 782000 nM T38200 CJ7P8C 70691309 IC50 = 3233000 nM T38200 C53QGB 118711599 IC50 = 76300 nM T38200 CO18BS 137635197 IC50 = 405000 nM T38200 CQL64H 137637846 IC50 > 1000000 nM T38200 CZ73DV 137638595 IC50 > 100000 nM T38200 CARI53 137638617 IC50 > 100000 nM T38200 CUM2T0 137638836 IC50 > 100000 nM T38200 C3PY5G 137638838 IC50 > 50000 nM T38200 CP7OV5 137639241 IC50 > 100000 nM T38200 C21IZT 137639281 IC50 > 1000000 nM T38200 CP24OX 137642163 IC50 > 100000 nM T38200 CK2VU3 137650102 IC50 > 1000000 nM T38200 C52PYO 137650910 IC50 > 1000000 nM T38200 CS6FX4 137651374 IC50 > 1000000 nM T38200 CPLJ94 137651669 IC50 > 1000000 nM T38200 CN04QK 137652511 IC50 > 1000000 nM T38200 CGC1Z4 137654858 IC50 > 50000 nM T38200 CADN74 137657292 IC50 > 100000 nM T38200 C4NK1W 137658990 IC50 > 50000 nM T38200 CPI4S8 137659917 IC50 > 50000 nM T38200 CI7S8H 155516242 IC50 > 100000 nM T38200 CL2TZ4 155518880 IC50 = 2754.23 nM T38200 C4U8QT 155524561 IC50 > 100000 nM T38200 CJ4OV6 155530359 IC50 > 100000 nM T38200 C4RL9X 155535776 IC50 > 100000 nM T38200 C7XS6Z 155549186 IC50 = 9332.54 nM T38200 CL2Q6G 155567178 IC50 > 100000 nM T38200 D02ANG 5216267 IC50 = 125892.54 nM T38200 D03IWW 6575389 IC50 = 2320000 nM T38200 D08YGM 92409 IC50 = 944000 nM T38200 D0D2EF 1796510 IC50 = 51000 nM T38200 D0H7WK 10458835 IC50 = 5000 nM T38200 D0P3KI 9888030 IC50 = 8920 nM T38200 D0RF2M 4498 IC50 = 106000 nM T38200 D0V5OY 16725912 Ki > 100000 nM T38200 D0V7RG 3532 IC50 = 110000 nM T38200 D0W8SX 239 IC50 = 41200 nM T38200 D0X3CF 442879 IC50 > 500000 nM T29355 D02VTV 117968550 EC50 = 1100 nM T29355 D03LZO 117967861 EC50 = 4400 nM T29355 C70QRI 1026354 IC50 = 64000 nM T29355 CJF29V 2965792 IC50 = 46500 nM T29355 CJ4ID2 3718032 IC50 = 38000 nM T29355 CBX8T9 16451230 IC50 > 200000 nM T29355 C85NAQ 24858111 EC50 = 900 nM T29355 CM4J7H 44379494 EC50 = 36000 nM T29355 CPL71I 54596764 IC50 > 100000 nM T29355 CER5F1 67466175 IC50 > 100000 nM T29355 CYB1U4 76318201 IC50 = 2800 nM T29355 CVM64R 117967504 EC50 = 1400 nM T29355 CJY5W0 117967660 EC50 = 6800 nM T29355 C9F3YV 117967663 EC50 = 1000 nM T29355 CM5N2A 117967691 EC50 = 3400 nM T29355 C2G4ND 117967705 EC50 = 1200 nM T29355 CY1V9T 117976066 EC50 = 4900 nM T29355 CY2R4J 117976176 EC50 = 300 nM T29355 CGQ82T 118732749 IC50 = 50000 nM T29355 CIZF42 122178085 IC50 > 50000 nM T29355 CR53MN 122186750 EC50 = 3000 nM T29355 CX3NU8 122186767 EC50 = 4000 nM T29355 CEW2X8 122186780 EC50 = 2100 nM T29355 C6G0CZ 122580323 EC50 = 1600 nM T29355 CU50GO 134154293 IC50 = 41000 nM T29355 CL0WR7 134386479 EC50 = 5400 nM T29355 C6GC0O 137028680 EC50 = 6200 nM T29355 CWMH49 137638632 EC50 = 1900 nM T29355 C05DFP 137653852 EC50 = 2100 nM T29355 C8LEV4 139267760 IC50 = 7600 nM T29355 CUVO30 155515610 EC50 = 2400 nM T29355 CX5G9E 155528619 EC50 = 5200 nM T29355 CS3PF1 155533577 EC50 = 4600 nM T29355 CRH9J5 155534178 EC50 = 5100 nM T29355 CAE51Q 155534378 EC50 = 4800 nM T29355 C29RHJ 155544579 EC50 = 5400 nM T29355 CIN57Q 155556138 IC50 = 74000 nM T29355 CB8SD4 155557649 EC50 = 8700 nM T29355 C0BU1J 155560963 EC50 = 5400 nM T29355 D02TVQ 71268957 IC50 > 100000 nM T29355 D09CLP 439155 IC50 > 50000 nM T01092 D05ROI 44462760 IC50 = 53200 nM T01092 D0H0EQ 24826799 IC50 = 12 nM T01092 D0W5HK 216239 IC50 = 1500 nM T01092 D02XNW 5494449 IC50 = 208 nM T01092 D0LQ3L 77108121 IC50 = 0.4 nM T01092 C09BCS 23578 Ki = 63.1 nM T01092 C76XNU 643953 IC50 = 754 nM T01092 C5IOS0 670041 EC50 = 4100 nM T01092 C7X5WE 2828334 EC50 = 182 nM T01092 C86MXJ 3063662 IC50 = 794 nM T01092 CDLJ02 3078467 IC50 = 2000 nM T01092 C8B3WY 3078469 IC50 = 2000 nM T01092 CMV76B 3078470 IC50 = 10 nM T01092 CYE04H 3078480 IC50 = 1.6 nM T01092 CZ4WV2 3670283 IC50 = 126 nM T01092 CA82YG 4628569 EC50 > 10000 nM T01092 CL70MG 4634732 EC50 = 457 nM T01092 C7TA9J 10113568 Ki = 2.042 nM T01092 CIV15Q 10113978 IC50 = 873 nM T01092 CFB81R 10317604 IC50 = 160 nM T01092 CF8Q2B 11288934 EC50 = 18 nM T01092 C8ET0Q 12791776 IC50 > 10000 nM T01092 CD2E5U 13142332 EC50 > 10000 nM T01092 C4V0BX 20895670 IC50 = 79 nM T01092 C25UKC 21081761 IC50 = 1500 nM T01092 CSFK63 23646936 IC50 = 32 nM T01092 CJ5H1Z 23646938 IC50 = 10 nM T01092 CIP7T2 23646939 IC50 = 2500 nM T01092 CI32JB 23646942 IC50 = 100 nM T01092 CX30ZW 25023828 IC50 = 73.6 nM T01092 C38PUJ 45271185 IC50 = 600 nM T01092 CS9T8F 53466952 IC50 = 61 nM T01092 C0HY3M 53467389 IC50 = 58 nM T01092 CLP04A 53467390 IC50 = 14 nM T01092 CV7C0D 53469060 IC50 = 69 nM T01092 CY04AP 53469630 IC50 = 56 nM T01092 CU4B0V 53469825 IC50 = 116 nM T01092 C5B4NV 55157876 EC50 = 1077 nM T01092 CKFP29 57971132 IC50 = 13 nM T01092 CUB9N0 60236671 EC50 = 378 nM T01092 CD8AV0 60698388 IC50 > 10000 nM T01092 CXIQ15 60723604 IC50 = 316 nM T01092 CVY1Z2 62679367 EC50 > 10000 nM T01092 CX30KT 62679368 EC50 = 8562 nM T01092 COQ08Y 62679370 EC50 = 1233 nM T01092 C9DYZ5 71816195 IC50 = 630 nM T01092 CY8O3K 72724969 IC50 = 20 nM T01092 CW7YD6 72725026 IC50 = 16 nM T01092 C5SQ7I 72725027 IC50 = 32 nM T01092 CFB69C 72725028 IC50 = 10 nM T01092 CE7G9T 72725029 IC50 = 4 nM T01092 CFR80L 72725083 IC50 = 160 nM T01092 COP05E 76310255 IC50 = 10 nM T01092 CHB93K 76313942 IC50 = 200 nM T01092 CCS63Z 76317480 IC50 = 40 nM T01092 CL0BO7 76317481 IC50 = 320 nM T01092 CFYP81 76317482 IC50 = 32 nM T01092 CFX5S0 76321210 IC50 = 4000 nM T01092 C7SD8Z 76321211 IC50 = 500 nM T01092 CKD2R6 76321212 IC50 = 63 nM T01092 C9X6CZ 76321213 IC50 = 160 nM T01092 C1EMH2 76321214 IC50 = 10 nM T01092 CW95IP 76324828 IC50 = 160 nM T01092 C35VHG 76328382 IC50 = 320 nM T01092 CUB91G 76328383 IC50 = 10 nM T01092 CAD50N 76328384 IC50 = 16 nM T01092 C4MT3A 76332057 IC50 = 25 nM T01092 C9IC1L 76332058 IC50 = 3200 nM T01092 C0K5MP 76332059 IC50 = 6.3 nM T01092 CO7J2V 76332061 IC50 = 16 nM T01092 CE09XW 76335674 IC50 = 200 nM T01092 CPUD78 77230897 IC50 = 1030 nM T01092 CB5H7C 82244347 IC50 > 10000 nM T01092 CC0US3 90345286 IC50 = 7.9 nM T01092 CM73SR 90345378 IC50 = 0.94 nM T01092 CNTP05 90345427 IC50 = 50 nM T01092 CS43ZG 90351311 Ki = 0.8 nM T01092 CR9ZV7 90351952 IC50 = 0.5 nM T01092 C4LT3Y 91885439 IC50 = 8.6 nM T01092 C28GLZ 110728326 IC50 > 1000 nM T01092 CF20OX 118557066 IC50 = 5 nM T01092 C6V5XY 118557110 IC50 = 0.4 nM T01092 C5ZQ4I 118557139 IC50 = 0.79 nM T01092 C78DEX 118557145 IC50 = 1600 nM T01092 C98CAG 118557162 IC50 = 0.4 nM T01092 CFJ27P 118557220 IC50 = 400 nM T01092 CSJR15 118557245 IC50 = 79 nM T01092 C21IGS 118557254 IC50 = 320 nM T01092 C3LR2H 118557293 IC50 = 1.6 nM T01092 CCYI79 118557322 IC50 = 0.79 nM T01092 CSD2H6 118557338 IC50 = 3.2 nM T01092 C5O4ZV 118557362 IC50 = 0.079 nM T01092 C6S0NT 118557462 IC50 = 63 nM T01092 CE8J7H 118557468 IC50 = 25 nM T01092 C02OGI 118557491 IC50 = 1 nM T01092 C42EMA 118557502 IC50 = 0.5 nM T01092 C12PXU 118557507 IC50 = 0.5 nM T01092 CS6JK9 118557559 IC50 = 794 nM T01092 CU7I5M 118564393 IC50 = 200 nM T01092 C2U3FR 118564396 IC50 = 32 nM T01092 CU0DW4 118564398 IC50 = 5 nM T01092 C7TBH3 118564402 IC50 = 0.32 nM T01092 C3KNZ5 121439991 EC50 = 28 nM T01092 CCX27F 121440014 EC50 = 74 nM T01092 CUR74H 121440015 EC50 > 3000 nM T01092 CH3CO4 121440032 EC50 = 262 nM T01092 CE0QC9 121440033 EC50 = 49 nM T01092 CJ0A5S 121440051 EC50 = 64 nM T01092 CLJI17 121446658 EC50 = 628 nM T01092 CY5A1S 121446659 EC50 = 125 nM T01092 C0HFX3 121446661 EC50 > 10000 nM T01092 C04IQZ 121446667 EC50 > 3000 nM T01092 C19DEL 121446676 EC50 = 490 nM T01092 C4FAO7 121446682 EC50 = 1234 nM T01092 CKUM01 121446684 EC50 = 56 nM T01092 CTM6K0 121446695 EC50 > 3000 nM T01092 CY61UA 121446710 EC50 = 1526 nM T01092 CWN4T7 121446721 EC50 = 1735 nM T01092 C0ZE8M 121446729 EC50 > 10000 nM T01092 CTXO48 121446730 EC50 = 898 nM T01092 C57TND 121446732 EC50 = 1254 nM T01092 CQH48Z 121446733 EC50 > 10000 nM T01092 CYTZ27 121446735 EC50 > 10000 nM T01092 C1ENL2 121446737 EC50 > 10000 nM T01092 CH68FX 121446738 EC50 = 221 nM T01092 C8SK7Y 121446739 EC50 = 628 nM T01092 C54DCI 121446741 EC50 > 10000 nM T01092 C1K5ZD 121446742 EC50 > 5000 nM T01092 CO32FQ 121446750 EC50 > 10000 nM T01092 C1FU2G 121446752 EC50 > 10000 nM T01092 CJ08HW 121446757 EC50 = 627 nM T01092 CX06JV 121446760 EC50 = 2527 nM T01092 C2ZF7V 121446761 EC50 = 8237 nM T01092 CB3I0L 121446764 EC50 = 656 nM T01092 C1H3VY 121446771 EC50 = 1308 nM T01092 C0B1WO 121446775 EC50 = 198 nM T01092 CU92HQ 121446778 EC50 = 58 nM T01092 C08KJZ 121446782 EC50 = 72 nM T01092 CVM06Q 121446783 EC50 = 36 nM T01092 CCD94Y 121446786 EC50 > 10000 nM T01092 CT8K2N 121446791 EC50 > 10000 nM T01092 C4NT5D 121446843 EC50 > 3000 nM T01092 CGP13F 121446847 EC50 = 12 nM T01092 CNH04D 121446878 EC50 = 98 nM T01092 C4QV9N 121446902 EC50 = 815 nM T01092 C8P4AE 122703561 IC50 = 10 nM T01092 C9E5DT 122703570 IC50 = 2 nM T01092 CM7C5F 122703576 IC50 = 7.9 nM T01092 CF5WY1 122703578 IC50 = 10 nM T01092 CF4PR9 122703579 IC50 = 16 nM T01092 C74SQF 122703581 IC50 = 13 nM T01092 CPA2Z5 122703584 IC50 = 10 nM T01092 CW70QA 122703585 IC50 = 63 nM T01092 CA6Z5C 122703586 IC50 = 10 nM T01092 CYIP81 122703588 IC50 = 10 nM T01092 C5LYJ9 122703599 IC50 = 126 nM T01092 CL7MB6 122703611 IC50 = 16 nM T01092 CJ3RT5 122703613 IC50 = 1.6 nM T01092 C6NT4C 122703637 IC50 = 10 nM T01092 C2TE3N 122703644 IC50 = 9 nM T01092 CP31IH 122703646 IC50 = 200 nM T01092 CIA2M8 122703656 IC50 = 6.3 nM T01092 CX7BC0 122703665 IC50 = 4 nM T01092 CKY5L7 122703666 IC50 = 316 nM T01092 C6R7MN 122703671 IC50 = 10 nM T01092 CAEG59 122703680 IC50 = 10 nM T01092 C8ODW1 122703682 IC50 = 10 nM T01092 CXA83K 122703688 IC50 > 10000 nM T01092 CR1C5H 122703691 IC50 = 4.8 nM T01092 CU7TI5 122703692 IC50 = 10 nM T01092 C27BKA 122703700 IC50 = 1.6 nM T01092 C26JOL 122703705 IC50 = 10 nM T01092 CR75IM 122703716 IC50 = 10 nM T01092 CEG87H 122703723 IC50 = 10 nM T01092 CG7RC6 122703734 IC50 = 398 nM T01092 CK2D8E 122703743 IC50 = 0.5 nM T01092 CZ6R3X 124086061 IC50 = 35 nM T01092 C9XVO7 124086067 IC50 = 10 nM T01092 C7MLB2 124086077 IC50 = 16 nM T01092 CJXY94 124180534 IC50 = 32 nM T01092 CY8JW7 127033346 IC50 > 10000 nM T01092 C3ASY7 127033640 IC50 = 35 nM T01092 C4BKW6 127033641 IC50 = 210 nM T01092 C1KNJ3 127033642 IC50 = 0.2 nM T01092 C1U6TC 130299179 IC50 = 631 nM T01092 C6IZ3V 130299401 IC50 = 3162 nM T01092 CNI1W2 132016672 IC50 = 79 nM T01092 CPF5E3 132471860 Ki = 0.912 nM T01092 CK4HX5 134521326 IC50 = 10 nM T01092 CRT5O7 134521520 IC50 = 8.5 nM T01092 C2E7AT 134521814 IC50 = 1 nM T01092 CG9R3J 134522007 IC50 = 10 nM T01092 CZB75S 134522265 IC50 = 2.5 nM T01092 CSCT10 134536604 IC50 = 7.9 nM T01092 CSL60X 135308861 Ki = 0.912 nM T01092 C0ZQP5 135308877 Ki = 1.738 nM T01092 CS1DF9 135308888 Ki = 13.8 nM T01092 CFX4W3 135308904 Ki = 251.19 nM T01092 CNF6O4 135308906 Ki = 1.778 nM T01092 C6M9FG 135308913 Ki = 2.57 nM T01092 CF1LY8 135308922 Ki = 6918.31 nM T01092 C3XG8C 135308924 Ki = 2.512 nM T01092 C8Z7AU 135308925 Ki = 1.148 nM T01092 C6EW1J 135308927 Ki = 3.467 nM T01092 C8NC5R 135308928 Ki = 2.951 nM T01092 C2C5TL 135308931 Ki = 4265.8 nM T01092 CZP1T3 135308934 Ki = 5.129 nM T01092 CNI5C3 135308946 Ki = 38.02 nM T01092 C8AVZ0 135308996 Ki = 3.89 nM T01092 CSOZ57 135309005 Ki = 7.943 nM T01092 CGFM04 135309027 Ki = 117.49 nM T01092 CQIU03 135309039 Ki = 107.15 nM T01092 CRJ8H5 135309049 Ki = 54.95 nM T01092 C5GAV8 135309066 Ki = 0.8511 nM T01092 CZ53KU 135309069 Ki = 33.88 nM T01092 CA28GI 135309090 Ki = 0.4074 nM T01092 CI8Z2F 135309102 Ki = 1.148 nM T01092 C5E6UB 135314480 IC50 = 39.81 nM T01092 CXC69T 137321158 IC50 = 11 nM T01092 CVGN14 137632484 IC50 = 0.05 nM T01092 C8PV3G 137632977 IC50 > 10000 nM T01092 COL6Q7 137634539 IC50 = 12600 nM T01092 C1FTS9 137634957 IC50 > 10000 nM T01092 C5KYE7 137635049 IC50 = 100 nM T01092 C3EIS6 137635629 IC50 = 0.4 nM T01092 CA8GF2 137637401 IC50 = 2468 nM T01092 CQ32NB 137638108 EC50 > 10000 nM T01092 C58MXE 137640092 IC50 = 2 nM T01092 C5B9NR 137640099 IC50 = 501 nM T01092 CZS13Q 137640111 IC50 = 295 nM T01092 C62DVJ 137640435 EC50 > 3000 nM T01092 CGC9T1 137641614 IC50 > 10000 nM T01092 CESF45 137644276 IC50 = 167 nM T01092 C4TBJ8 137647324 IC50 > 10000 nM T01092 CLP5H9 137647405 IC50 = 0.63 nM T01092 C4JH8A 137647835 IC50 > 10000 nM T01092 CYP70I 137651336 IC50 > 10000 nM T01092 CCK03W 137652965 IC50 > 10000 nM T01092 CKX2D8 137654471 IC50 > 10000 nM T01092 CRH18Z 137656846 IC50 = 178 nM T01092 CP51KG 137657894 IC50 = 1259 nM T01092 CFH52E 137659234 IC50 = 251 nM T01092 C3BCN1 138377545 IC50 = 0.3 nM T01092 CGX92C 138393291 IC50 = 5500 nM T01092 CCT23N 141340950 IC50 > 15000 nM T01092 CTS9Q8 142416001 IC50 = 2.512 nM T01092 CFGH25 142416011 IC50 = 10 nM T01092 C2X1CR 145978863 IC50 = 190 nM T01092 C85UBM 145978937 IC50 = 10 nM T01092 CAW7B1 145980780 IC50 = 468 nM T01092 C43ZUJ 145981140 IC50 = 49 nM T01092 C10HDT 145981335 IC50 = 134 nM T01092 C8DKN3 145981423 IC50 = 94 nM T01092 C89BNR 145982306 IC50 = 531 nM T01092 CO57FT 145982439 IC50 = 3457 nM T01092 CUZQ37 145985171 IC50 = 704 nM T01092 C41ZBR 145986358 IC50 = 105 nM T01092 C4D8HB 145986929 IC50 = 18 nM T01092 C3FN9P 145987011 IC50 = 424 nM T01092 CST1O6 145987202 IC50 = 31 nM T01092 CGM18W 145987557 IC50 = 10 nM T01092 CAC0M7 145988480 IC50 = 13 nM T01092 C7DWU4 145988653 IC50 = 26 nM T01092 CUJL09 145988701 IC50 = 77 nM T01092 C58ULD 145988885 IC50 = 49 nM T01092 CVH28K 145989341 IC50 = 128 nM T01092 COTX64 145989416 IC50 = 2994 nM T01092 C8VND5 145989851 IC50 = 10 nM T01092 C4P8HQ 145990145 IC50 = 264 nM T01092 CZ0RI5 145990208 IC50 = 107 nM T01092 CGF6E4 145990858 IC50 = 17 nM T01092 C96XWF 145991904 IC50 = 28 nM T01092 C3D6OB 145992043 IC50 = 79 nM T01092 CAOQ30 145992060 IC50 = 392 nM T01092 C1NYL4 145993423 IC50 = 634 nM T01092 C05WAM 146344085 IC50 = 90 nM T01092 CN7MS2 154023591 IC50 = 5 nM T01092 CKW68P 155393270 IC50 = 7940 nM T01092 CS0T6E 155510707 IC50 = 17000 nM T01092 C37FPZ 155510738 IC50 > 15000 nM T01092 CX0T1C 155512182 IC50 = 10 nM T01092 C0AUE4 155512296 IC50 = 10 nM T01092 COA84W 155512492 IC50 = 200 nM T01092 C23DJP 155512860 IC50 = 19.95 nM T01092 C2MD1Q 155513187 IC50 > 10000 nM T01092 CZ7K6H 155513660 IC50 > 15000 nM T01092 CC3T0M 155518699 IC50 = 10 nM T01092 CWZ5J8 155519113 IC50 = 5012 nM T01092 CXD9M4 155520427 IC50 = 10 nM T01092 C4FW0B 155522577 IC50 = 6.3 nM T01092 CLW39S 155522794 IC50 = 10 nM T01092 CQIR50 155523679 IC50 = 200 nM T01092 C9M2ZT 155523831 IC50 = 10 nM T01092 CPK67I 155524868 IC50 = 180 nM T01092 CJ3M5T 155524881 IC50 > 1000 nM T01092 CU9H3G 155525351 Ki = 21 nM T01092 C1ICR3 155529856 IC50 > 10000 nM T01092 CIP84Q 155530191 IC50 = 90 nM T01092 C0V9QN 155532882 IC50 > 15000 nM T01092 CTJ84E 155533767 IC50 = 1.3 nM T01092 CQOE59 155534156 IC50 = 310 nM T01092 CF09IN 155535999 IC50 = 10 nM T01092 C8JR2S 155537020 IC50 = 20.8 nM T01092 CSU48D 155537554 IC50 = 10 nM T01092 CZR0J9 155537757 IC50 = 11000 nM T01092 CTP72E 155538424 IC50 = 200 nM T01092 CZ80HO 155547269 IC50 = 10 nM T01092 CSQ28H 155548887 IC50 = 2.5 nM T01092 C5L7HY 155551127 IC50 > 15000 nM T01092 CQ92XF 155552769 IC50 = 126 nM T01092 CDT06B 155555771 IC50 = 600 nM T01092 CL2CH8 155556595 IC50 = 10 nM T01092 C4Z8UW 155569299 IC50 = 1.3 nM T01092 D0K8YD 76332060 IC50 = 16 nM T01092 D0N4LR 53469448 IC50 = 18 nM T99149 D04XVN 11707110 IC50 = 1.6 nM T99149 D0E3TC 44259 IC50 = 37.4 nM T99149 D0K0YC 9826528 IC50 = 110 nM T99149 D0A9KI 9863367 IC50 > 50 nM T99149 C8KED5 4713 IC50 = 50000 nM T99149 CQ7PL4 1235170 IC50 > 20000 nM T99149 C5VPH9 16129448 IC50 = 391 nM T99149 C0H8UN 16730109 IC50 > 30000 nM T99149 C6P1CX 25066843 IC50 > 20000 nM T99149 C3VRO9 44557921 IC50 > 10000 nM T99149 CIPX17 45485590 Ki = 9700 nM T99149 CI10RQ 45485600 Ki = 13000 nM T99149 CPVU61 45485609 Ki = 6200 nM T99149 C58VXQ 45485625 Ki = 710 nM T99149 CMI83V 45485640 Ki = 2400 nM T99149 CP87FU 45485645 Ki = 1400 nM T99149 CLJF04 45485646 Ki = 1800 nM T99149 CQE7Z0 45485654 Ki = 3700 nM T99149 C5J4CW 45485664 Ki = 1400 nM T99149 C63VLU 45485665 Ki = 1800 nM T99149 C7VRC1 45485666 Ki = 2100 nM T99149 CK8Q9R 45485676 Ki = 16000 nM T99149 C7SX0U 45485677 Ki = 670 nM T99149 C4UB6E 45485687 Ki = 1400 nM T99149 CRA74I 49842779 IC50 = 6840 nM T99149 C37NKO 67129970 IC50 > 10000 nM T99149 CK80LJ 67130050 IC50 > 10000 nM T99149 CV63UL 67240318 IC50 > 10000 nM T99149 C7GRV2 68755406 IC50 > 10000 nM T99149 C2LAM7 126591927 IC50 = 82 nM T99149 CI2YE9 132606873 IC50 = 186.7 nM T99149 C0TE5S 135651612 IC50 = 1300 nM T99149 CI1E8V 137634241 IC50 > 10000 nM T99149 CU62AO 145712394 IC50 = 590 nM T99149 C6VB3O 145925651 IC50 >= 5000 nM T99149 C2MD1Q 155513187 IC50 > 10000 nM T99149 C4NKP6 155518298 IC50 = 1500 nM T99149 C86HPW 155518524 IC50 = 74000 nM T99149 D08LYB 5166 IC50 > 50 nM T99149 D0GD8Y 3006531 IC50 = 58 nM T48780 CZ7HO2 24139 IC50 = 125892.54 nM T48780 CSO4E3 644170 IC50 = 1000000000 nM T48780 C0FSW1 2733653 IC50 = 4.3 nM T48780 CDPK78 7177184 IC50 = 1000000000 nM T48780 CNC34Y 11182549 IC50 = 0.5012 nM T48780 C7HF4C 13018787 IC50 = 630957.34 nM T48780 CD7TM6 15423759 IC50 = 398107.17 nM T48780 C90UTG 15471714 IC50 = 12.59 nM T48780 CUB5A3 16182677 IC50 = 63.1 nM T48780 C3TJZ4 46233136 IC50 = 14 nM T48780 CRK14X 46233137 IC50 = 251188.64 nM T48780 CXYW80 46233138 IC50 = 79432.82 nM T48780 C0EO5S 46233140 IC50 = 79.43 nM T48780 CZ7UL4 46233142 IC50 = 31622.78 nM T48780 C8ZC9X 49798491 IC50 = 3981.07 nM T48780 CSRN46 49863275 IC50 = 501187.23 nM T48780 CQT6X8 49863277 IC50 = 31622.78 nM T19531 C71SIH 253167 IC50 > 200000 nM T19531 CWC34Q 259205 IC50 > 200000 nM T19531 C8QM7B 6852376 EC50 = 80 nM T19531 CAD72T 9817518 IC50 = 10800 nM T19531 CZTH29 9834991 IC50 = 78000 nM T19531 CR52JI 9910619 IC50 = 7.2 nM T19531 CB3I8J 10014327 IC50 = 7900 nM T19531 CXZ8F3 10469457 IC50 = 13600 nM T19531 C2FP5Q 10617830 IC50 > 200000 nM T19531 CXMT71 10858184 IC50 > 200000 nM T19531 CA2ZN5 10869068 IC50 = 4600 nM T19531 CUM3X1 10912229 IC50 > 200000 nM T19531 C3VSN6 10912305 IC50 = 200 nM T19531 CQ4J5L 10934245 IC50 > 100000 nM T19531 CTX59A 10934704 IC50 = 600 nM T19531 C51JOG 10945208 IC50 > 200000 nM T19531 CQ45ND 10956699 IC50 = 16300 nM T19531 C72IAN 10989023 IC50 = 4900 nM T19531 CC4K0Z 10989442 IC50 = 400 nM T19531 CR7VM3 11000246 IC50 = 2600 nM T19531 CL06OV 11021644 IC50 > 200000 nM T19531 C8IO0S 11032616 IC50 = 188000 nM T19531 CM5XW9 11043528 IC50 = 28800 nM T19531 CK0IO4 11054944 IC50 = 55000 nM T19531 C3TOQ4 11086961 IC50 = 4300 nM T19531 CH91TK 11097296 IC50 = 100000 nM T19531 C7OTX5 11108129 IC50 > 70000 nM T19531 C5I0MZ 11139808 IC50 = 8200 nM T19531 C3NEH9 11776872 IC50 = 7600 nM T19531 CN4SE5 11780214 IC50 = 73200 nM T19531 CIX40T 11780786 IC50 = 9400 nM T19531 CUVM56 11832149 IC50 > 200000 nM T19531 C4R9QU 11832661 IC50 = 25100 nM T19531 CTM46O 14787969 EC50 = 210 nM T19531 CS6BV5 44309263 IC50 = 35400 nM T19531 CPA3N4 44335158 IC50 > 200000 nM T19531 CZM7L2 44335253 IC50 > 200000 nM T19531 CC5D0B 44335255 IC50 > 200000 nM T19531 CS75WN 44335277 IC50 > 200000 nM T19531 CCH3Y5 44335278 IC50 = 15300 nM T19531 CX7S8F 44335279 IC50 > 200000 nM T19531 CAQ09P 44335291 IC50 > 200000 nM T19531 C73QWO 44335292 IC50 > 200000 nM T19531 C2DX5B 44335293 IC50 > 200000 nM T19531 C8RME2 44335295 IC50 > 200000 nM T19531 CEY06B 44335296 IC50 > 200000 nM T19531 CV51XU 44335303 IC50 > 200000 nM T19531 COHV64 44335304 IC50 > 200000 nM T19531 C3T8LU 44335305 IC50 > 200000 nM T19531 CXT80K 44335306 IC50 > 200000 nM T19531 CB2HR3 44335308 IC50 > 200000 nM T19531 C2VU5P 44335316 IC50 > 200000 nM T19531 CLJ93K 44335335 IC50 = 140500 nM T19531 C60VLZ 44335352 IC50 > 200000 nM T19531 C47QRL 44335393 IC50 = 94000 nM T19531 C84RSA 44335432 IC50 > 200000 nM T19531 CCJB21 44335433 IC50 > 200000 nM T19531 CU25TG 44335465 IC50 > 200000 nM T19531 C1Y6QO 44335470 IC50 > 200000 nM T19531 C2JTN3 44335685 IC50 > 200000 nM T19531 CLK79Y 44335691 IC50 > 200000 nM T19531 C93OIU 44335698 IC50 > 200000 nM T19531 CIGM53 44335700 IC50 = 72000 nM T19531 C3MWY8 44335701 IC50 = 110000 nM T19531 CF7MS0 44335709 IC50 = 13600 nM T19531 CY8E2J 44335711 IC50 > 200000 nM T19531 CH5J4P 44335712 IC50 = 78000 nM T19531 CI4R0U 44335725 IC50 = 79000 nM T19531 CD7LE2 44335742 IC50 = 102000 nM T19531 C68TLS 44335939 IC50 = 98000 nM T19531 CGBF56 44335982 IC50 = 10800 nM T19531 C3NA5F 44461049 EC50 = 8 nM T97174 C13QNP 65127 IC50 = 23000 nM T97174 CAO2X9 25169386 IC50 = 150000 nM T97174 C5TBY8 25169388 IC50 = 71000 nM T97174 CVX2B3 25169390 IC50 = 22000 nM T97174 COXH93 44589903 IC50 = 230000 nM T31543 D05EAM 4735 Ki = 1160 nM T31543 D07XHO 4413 Ki = 0.02 nM T31543 D0KG3R 9875401 Ki = 3350 nM T31543 C2KE5Q 1508 Ki = 60000 nM T31543 CUSM50 11974 Ki = 535 nM T31543 C5P3TH 65130 Ki = 924 nM T31543 CZ1QL5 411406 Ki = 191 nM T31543 CB9VP7 432298 Ki = 200 nM T31543 C8VB4U 480183 Ki = 719 nM T31543 CROX25 480185 Ki = 397 nM T31543 CO5Y7H 725447 IC50 = 111000 nM T31543 CPJ28H 828532 IC50 = 420 nM T31543 CJ1GN3 869194 IC50 = 98000 nM T31543 CBFT53 975107 IC50 > 30000 nM T31543 CQUP23 2208579 IC50 = 75000 nM T31543 C97ZIP 2262135 IC50 = 120000 nM T31543 C74DMH 2262990 IC50 = 103000 nM T31543 CQPJ74 2938648 IC50 > 30000 nM T31543 C4S9WR 3000497 Ki = 816 nM T31543 C4Z0XK 3010932 Ki = 2280 nM T31543 C6WU4N 5000438 IC50 > 30000 nM T31543 CQ26VM 5289531 Ki = 170 nM T31543 CHY56L 5729350 IC50 = 138000 nM T31543 CI69XU 5739522 IC50 = 128000 nM T31543 CN2B6S 6852211 Ki = 4.3 nM T31543 CKDP84 9895193 Ki = 320 nM T31543 CDT95S 9939426 Ki = 370 nM T31543 CEC95B 9997816 Ki = 9600 nM T31543 CB1S5N 11363919 Ki = 7180 nM T31543 CJZ09N 11512593 Ki = 340 nM T31543 C28BMR 11513105 Ki = 13 nM T31543 CRNU10 11534959 Ki = 50 nM T31543 CD1A6T 11542037 Ki = 61 nM T31543 CA8KD7 11542038 Ki = 65 nM T31543 CBP69L 11557024 Ki = 1.8 nM T31543 CCG84F 11563457 Ki = 89 nM T31543 CV46NL 11563632 Ki = 730 nM T31543 CEAZ46 11569930 Ki = 160 nM T31543 C3TJ7M 11570580 Ki = 88 nM T31543 C6RHD8 11570700 Ki = 1.5 nM T31543 C1DN2L 11570759 Ki = 690 nM T31543 C6FG8V 11577055 Ki = 110 nM T31543 CIY34V 11577968 Ki = 200 nM T31543 CJ38EP 11577970 Ki = 690 nM T31543 C7MF9N 11578158 Ki = 89 nM T31543 CTSK74 11584729 Ki = 3.8 nM T31543 C1RQ6P 11592130 Ki = 3.9 nM T31543 CBC84M 11592593 Ki = 140 nM T31543 C7ZS8L 11592600 Ki = 44 nM T31543 C7QTY8 11606981 Ki = 4.2 nM T31543 CU07NO 11607091 Ki = 100 nM T31543 CL9TZ2 11614477 Ki = 140 nM T31543 CB4O2Q 11621579 Ki = 61 nM T31543 CD3R1E 11627899 Ki = 75 nM T31543 CB9P0Q 11628768 Ki = 8.7 nM T31543 CO3Q9N 11635973 Ki = 330 nM T31543 CRX98P 11636026 Ki = 53 nM T31543 CW10CL 11642802 Ki = 45 nM T31543 C2W5XF 11656797 Ki = 28 nM T31543 C4SAR0 11657278 Ki = 1500 nM T31543 CVQ16C 11664107 Ki = 42 nM T31543 CPZG49 11664334 Ki = 400 nM T31543 CT9E0G 11664643 Ki = 57 nM T31543 CWV87X 11671266 Ki = 5 nM T31543 CE0A6N 11671776 Ki = 96 nM T31543 C85GCY 11671956 Ki = 130 nM T31543 C1DHO6 11678360 Ki = 120 nM T31543 C4IBO3 11678764 Ki = 13 nM T31543 C69YSR 11693028 Ki = 380 nM T31543 CCQY30 11693049 Ki = 21 nM T31543 CPFW75 11699600 Ki = 72 nM T31543 C3VS2H 11699903 Ki = 53 nM T31543 CNV09Z 11699913 Ki = 38 nM T31543 CKQ4O2 11721188 Ki = 210 nM T31543 C4UB2X 11721375 Ki = 250 nM T31543 CRD97T 14477068 Ki > 10000 nM T31543 C1Z9SX 24776379 Ki = 200 nM T31543 CAO2V4 25030840 Ki = 7.5 nM T31543 CU82IO 25030929 Ki = 3 nM T31543 C7MCT6 25031099 Ki = 37 nM T31543 C5PO7A 25031100 Ki = 255 nM T31543 CH7Z1K 25031101 Ki = 12 nM T31543 CEW9X2 25031102 Ki = 6.1 nM T31543 C9NC4S 25031541 Ki = 33 nM T31543 CK5R8Q 25032200 Ki = 13 nM T31543 CG8HY2 25032202 Ki = 31 nM T31543 CH76XK 25032204 Ki = 65 nM T31543 CG76TR 25181493 Ki = 7 nM T31543 CA81RS 44144381 Ki = 220 nM T31543 CMZ05T 44324727 Ki = 40500 nM T31543 CE9I1R 44362422 Ki = 1800 nM T31543 CF5XO4 44413343 Ki = 84 nM T31543 CTD42X 44413355 Ki = 240 nM T31543 C9KQM2 44413356 Ki = 26 nM T31543 CQDX92 44413619 Ki = 100 nM T31543 CBSG69 44413636 Ki = 82 nM T31543 CU4AE5 44436348 Ki = 0.92 nM T31543 CVI26C 44436349 Ki = 4750 nM T31543 CZX07Q 44436350 Ki > 250000 nM T31543 C3X8OV 44436352 Ki = 90000 nM T31543 C9MOC3 44436353 Ki = 22500 nM T31543 CZF8M1 44436354 Ki = 28000 nM T31543 C3PGJ7 44436356 Ki = 107000 nM T31543 CRP6D7 44436357 Ki = 2330 nM T31543 CDI8A3 44436358 Ki = 450 nM T31543 C64FDS 44436359 Ki = 1000 nM T31543 C7PN9C 44436360 Ki = 890 nM T31543 C1RZ4Y 44436365 Ki = 857 nM T31543 CPEM68 44436366 Ki = 380 nM T31543 C8LQS9 44436368 Ki = 160 nM T31543 CEW6G1 44569299 Ki = 0.08 nM T31543 C9JNT3 44569300 Ki = 28 nM T31543 C9XE7Q 44569301 Ki = 56 nM T31543 CZI8D7 44569333 Ki = 2800 nM T31543 CK9YI3 44569356 Ki = 10000 nM T31543 C7XE6N 44569357 Ki > 1000000 nM T31543 C5ZG0T 44569358 Ki > 1000000 nM T31543 CR4CP6 44569359 Ki = 145 nM T31543 C9JF7W 44569667 Ki = 1 nM T31543 C61IJB 44569732 Ki = 6.7 nM T31543 CR36MB 44569733 Ki = 120 nM T31543 CE25UL 44569767 Ki = 180 nM T31543 C0CZ4I 44569768 Ki = 41 nM T31543 CIR4M0 44569769 Ki = 110 nM T31543 C02SHD 44569811 Ki = 29 nM T31543 CG3LE9 44569812 Ki = 91 nM T31543 CCU7V0 44569813 Ki = 26 nM T31543 C8BR6E 44569843 Ki = 6 nM T31543 C7Q9BH 44569844 Ki = 12 nM T31543 CZ35OW 44569845 Ki = 5.4 nM T31543 CHV9C1 44569846 Ki = 2.5 nM T31543 C5JQ4W 44569889 Ki = 60 nM T31543 CE1O4I 44569890 Ki = 47 nM T31543 C4JU7I 44569891 Ki = 13 nM T31543 CGS83Z 44569892 Ki = 1.6 nM T31543 C4BN3H 44573109 Ki = 6.3 nM T31543 COR57Y 44573272 Ki = 53 nM T31543 C6DX3Y 44573273 Ki = 17 nM T31543 CM2R1P 44573274 Ki = 53 nM T31543 CSP1I0 44573310 Ki = 150 nM T31543 C6EG9V 44573311 Ki = 180 nM T31543 CYV3X2 44573378 Ki = 470 nM T31543 CWUA41 44573379 Ki = 100 nM T31543 CYA64G 44573380 Ki = 2400 nM T31543 CLG42S 44573428 Ki = 11000 nM T31543 C4RSI0 46899736 Ki = 770 nM T31543 CX0Y2G 46899738 Ki = 2100 nM T31543 CLC94G 46918674 Ki = 972.9 nM T31543 C54AGL 46918753 Ki = 1710.7 nM T31543 CG7K0O 46937165 Ki = 457 nM T31543 CXUM36 49820499 Ki = 200 nM T31543 CX7SA8 49820500 Ki = 40 nM T31543 CQ3R6L 49820501 Ki = 200 nM T31543 CSFD83 49820654 Ki = 1200 nM T31543 CS8FY6 49820655 Ki = 545 nM T31543 C6OIW8 49820657 Ki = 600 nM T31543 CJ5G9Q 49820816 Ki = 1131 nM T31543 CL8UV3 49820969 Ki = 40 nM T31543 C2B5EC 49820973 Ki = 301 nM T31543 CAM3V7 50939649 Ki = 2 nM T31543 CHC74O 50939651 Ki = 23 nM T31543 CSAQ19 66818162 Ki = 40 nM T31543 COAY94 66818433 Ki = 1790 nM T31543 CG9UM3 66818450 Ki = 141 nM T31543 CG0TZ3 66818504 Ki = 1982 nM T31543 CU6E0A 66818541 Ki = 3 nM T31543 C89BXR 66818555 Ki = 400 nM T31543 C6LD2R 66818559 Ki = 10 nM T31543 C6CP8D 66818568 Ki = 6 nM T31543 CKD8I1 66818569 Ki = 10 nM T31543 C05LHZ 66818575 Ki = 592 nM T31543 CDA2M4 66818582 Ki = 1698 nM T31543 C9LTK3 66818589 Ki = 500 nM T31543 C9FQY8 66818629 Ki = 2032 nM T31543 C9GM3F 66818639 Ki = 260 nM T31543 C4U7SZ 66818677 Ki = 18 nM T31543 CL8D0V 66818717 Ki = 18 nM T31543 C41RKZ 66818743 Ki = 200 nM T31543 C6Q8FO 66818744 Ki = 411 nM T31543 CE53KG 66818763 Ki = 1060 nM T31543 CJA30C 66818765 Ki = 204 nM T31543 C5LU1Z 66818766 Ki = 1 nM T31543 CR94HZ 66818781 Ki = 1850 nM T31543 CP18VA 66818813 Ki = 770 nM T31543 CF4PT6 66818819 Ki = 824 nM T31543 CYB76J 66818882 Ki = 116 nM T31543 CRH5O7 66818889 Ki = 100 nM T31543 CGI6B3 66819113 Ki = 61 nM T31543 C4JV1L 66820910 Ki = 730 nM T31543 C62LDA 66821311 Ki = 94 nM T31543 CK59IZ 68788696 Ki = 1617 nM T31543 CGA3T2 68789018 Ki = 3 nM T31543 CC0J3V 68790735 Ki = 23 nM T31543 C5S0OC 70682854 Ki = 0.088 nM T31543 CUM4H3 70684929 Ki = 6124 nM T31543 CAU0K6 70689168 Ki = 9.5 nM T31543 C70YQU 70689169 Ki = 1.4 nM T31543 C47HLV 70689173 Ki = 4.6 nM T31543 CVD3W9 71495381 Ki = 13 nM T31543 CNVH43 71495466 Ki = 13 nM T31543 CA5N2S 71495467 Ki = 51 nM T31543 CQ98NY 71495468 Ki = 120 nM T31543 CE15GB 71495559 Ki = 130 nM T31543 CW1Y2L 71495560 Ki = 52 nM T31543 C5Q9BD 71495561 Ki = 33 nM T31543 C36MRI 71495659 Ki = 8 nM T31543 C7PDA9 71495660 Ki = 1 nM T31543 CF3C8E 71495661 Ki = 11 nM T31543 CECD13 71495765 Ki = 74 nM T31543 C7LXK1 71495766 Ki = 18 nM T31543 CKQ82B 71495974 Ki = 14 nM T31543 CSV38K 71495975 Ki = 56 nM T31543 C7QPA0 71495976 Ki = 35 nM T31543 CI4P9Z 71495977 Ki = 39 nM T31543 CE03BA 71496089 Ki = 8 nM T31543 CLO24G 71496201 Ki = 14 nM T31543 CIE7A6 71496202 Ki = 26 nM T31543 CAM0I4 71496204 Ki = 120 nM T31543 C5MVT3 76310068 Ki = 2900 nM T31543 CWZA05 76320988 Ki = 40 nM T31543 CV7IW5 87167024 Ki = 793 nM T31543 CMC3L7 89399327 Ki = 11 nM T31543 CJ6CN0 90644019 Ki = 591 nM T31543 CB8KY3 90644020 Ki = 1182 nM T31543 CB3Z7W 90644021 Ki = 0.08 nM T31543 C0G6SP 90644022 Ki = 305 nM T31543 CH3US6 90644023 Ki = 470 nM T31543 C1SAZ8 90666139 Ki = 49 nM T31543 C2ERV8 90666140 Ki = 7 nM T31543 CSO5R7 90666141 Ki = 12 nM T31543 C3F0PB 90666142 Ki = 23 nM T31543 CG1W0R 90666143 Ki = 17 nM T31543 CI3AX1 90666144 Ki = 1.8 nM T31543 C43YWM 90666145 Ki = 0.9 nM T31543 CT45NA 90666146 Ki = 2.7 nM T31543 C56KQL 90666147 Ki = 5.1 nM T31543 CA90QH 91827690 Ki = 530 nM T31543 C65TLW 101862198 Ki > 1000000 nM T31543 C46MSP 118542774 Ki = 1280 nM T31543 C20WBY 118542785 Ki = 830 nM T31543 CI65YK 118542879 Ki = 850 nM T31543 CEH93P 118542958 Ki = 580 nM T31543 CITU59 118548755 Ki = 470 nM T31543 CMF5R6 118548758 Ki = 280 nM T31543 C1IH2W 118548759 Ki = 810 nM T31543 C6LZQ3 118548760 Ki = 330 nM T31543 C62ZNW 118548761 Ki = 520 nM T31543 C3WQ9D 118548776 Ki = 1510 nM T31543 CU01RP 118548813 Ki = 350 nM T31543 CYUL31 118720337 Ki = 0.061 nM T31543 C4SUL9 118720338 Ki = 0.18 nM T31543 CP4F0X 118720339 Ki = 0.23 nM T31543 C0QI8C 118720340 Ki = 0.14 nM T31543 C6UG4N 118720341 Ki = 0.72 nM T31543 COFR38 118720342 Ki = 0.15 nM T31543 CA7O2K 118720343 Ki = 0.092 nM T31543 C3E7IH 118720344 Ki = 14.67 nM T31543 C9Z4AQ 118720345 Ki = 0.91 nM T31543 CKLU87 118720346 Ki = 0.45 nM T31543 C2NE9Q 118720347 Ki = 7.98 nM T31543 CS2G7Z 118720348 Ki = 31.54 nM T31543 CC2EV6 118720349 Ki = 3.22 nM T31543 CL28SC 118720350 Ki = 1.4 nM T31543 CF64QE 118720351 Ki = 0.89 nM T31543 C7NG3I 118721642 Ki = 0.92 nM T31543 CTV97I 118721643 Ki = 22 nM T31543 C1NS7F 118721644 Ki = 32 nM T31543 C3OCD1 118721645 Ki = 0.69 nM T31543 CQK2U8 118721646 Ki = 15 nM T31543 C4HB3G 118721647 Ki = 0.32 nM T31543 CNP30X 118721648 Ki = 9.2 nM T31543 CRPV34 118721649 Ki = 1.1 nM T31543 CU5KB2 118721650 Ki = 5.5 nM T31543 CJA76N 118721651 Ki = 58 nM T31543 CS3GX9 118721652 Ki = 104 nM T31543 C0Y9EU 118721653 Ki = 8.6 nM T31543 CJ4FI3 118721654 Ki = 3 nM T31543 CK2QX9 118721655 Ki = 12 nM T31543 C4UYE3 118721656 Ki = 5.8 nM T31543 CP9L7H 118721657 Ki = 8.7 nM T31543 C2MI1J 118721658 Ki = 69 nM T31543 CIPY54 118721659 Ki = 0.83 nM T31543 CSAZ58 118728084 Ki = 14900 nM T31543 C4K6HY 118729129 Ki = 1500 nM T31543 C4MX0T 118729130 Ki = 6700 nM T31543 CUC7N1 118729131 Ki = 620 nM T31543 C1KWF0 118729132 Ki = 760 nM T31543 CS7QD3 118729855 Ki = 300 nM T31543 CWK9I0 118729856 Ki = 2600 nM T31543 C73DSK 118729857 Ki = 1200 nM T31543 CM2E0V 118729858 Ki = 4600 nM T31543 C63TEA 118729859 Ki = 480 nM T31543 CPD68M 118729860 Ki = 2500 nM T31543 C3NK4O 121232387 Ki = 2100 nM T31543 C0IAV8 122182389 Ki = 558 nM T31543 CXT84D 122182390 Ki = 526 nM T31543 CG4LR5 122194707 Ki = 4400 nM T31543 CA6U5Q 122194708 Ki = 4800 nM T31543 CZ8CH4 122194709 Ki = 500 nM T31543 CLDC14 122194710 Ki = 1500 nM T31543 C6NGM7 122194711 Ki = 800 nM T31543 CR4CY8 122194712 Ki = 1100 nM T31543 COY83A 122535266 Ki = 0.13 nM T31543 CG5S2R 122535267 Ki = 0.65 nM T31543 CAI69W 123238067 Ki = 1540 nM T31543 C76BAD 123424620 Ki = 850 nM T31543 CA30BN 127033248 Ki = 48900 nM T31543 CO7PY0 127033521 Ki = 13500 nM T31543 CE0QZ4 127033522 Ki = 15400 nM T31543 C7ZIR9 127034099 Ki = 510 nM T31543 C1BWV2 127035672 Ki > 1000000 nM T31543 CVRY56 127036086 Ki > 1000000 nM T31543 C9B6LT 127037264 Ki > 1000000 nM T31543 C60HLK 127037469 Ki > 1000000 nM T31543 C90LJI 127045142 Ki = 492 nM T31543 CD06PE 134313025 Ki = 3.1 nM T31543 CH74VX 135435498 Ki = 4500 nM T31543 CX52AQ 137631869 Ki = 44 nM T31543 CMB40N 137632239 Ki = 28 nM T31543 CDN14Z 137635697 Ki = 48 nM T31543 CDQ62V 137637214 Ki = 40000 nM T31543 CV3I9R 137637849 Ki = 240 nM T31543 CI5VX9 137639355 Ki = 63 nM T31543 C2K8JV 137639385 Ki = 15000 nM T31543 C5PHM2 137640910 Ki = 71 nM T31543 CI3JQ8 137640977 Ki = 150 nM T31543 C3TZH7 137640998 Ki = 120 nM T31543 CQ7N3P 137642872 Ki = 19 nM T31543 CVTM59 137644771 Ki = 12 nM T31543 CA7F3M 137645031 Ki = 200 nM T31543 C51JAT 137646077 Ki = 26 nM T31543 C94KVB 137646622 Ki = 12000 nM T31543 C6G4RT 137647792 Ki = 20 nM T31543 C3P0CS 137648443 Ki = 1380 nM T31543 C30ZQS 137648450 Ki = 120 nM T31543 CS03HK 137648571 Ki = 4 nM T31543 C6Z7LI 137653508 Ki = 7 nM T31543 CC0OE6 137653752 Ki = 39 nM T31543 C6HKV9 137654166 Ki = 43 nM T31543 CNX46H 137654508 Ki = 50000 nM T31543 CZW3F6 137655661 Ki = 15000 nM T31543 CT6X1A 137657743 Ki = 34 nM T31543 C38KYF 137658118 Ki = 5.6 nM T31543 C0Z8RH 137658426 Ki = 51 nM T31543 CXEV32 137659374 Ki = 230 nM T31543 CAE43N 137659536 Ki = 34 nM T31543 C0SJX8 137661290 Ki = 20 nM T31543 CXZ3O7 137662143 Ki = 65 nM T31543 CUZ35A 138115400 IC50 = 25118.86 nM T31543 C0A3MI 145959466 IC50 > 50000 nM T31543 CJP64T 155510867 IC50 = 90 nM T31543 CZR36C 155511554 IC50 = 7943.28 nM T31543 CUP78D 155512098 IC50 = 640 nM T31543 CYT20V 155514020 Ki > 50000 nM T31543 C1RYT8 155517297 Ki = 486 nM T31543 C6NX4K 155519661 IC50 = 1995.26 nM T31543 C4MS1B 155519676 IC50 = 39810.72 nM T31543 CX6C5Y 155520312 IC50 = 4000 nM T31543 CE01NY 155523107 IC50 = 730 nM T31543 CW9K3R 155523263 IC50 = 1100 nM T31543 CGMP07 155523803 Ki = 0.55 nM T31543 CRC6L7 155524551 IC50 > 10000 nM T31543 C4HN6V 155525157 Ki = 271 nM T31543 C6L1WU 155525184 Ki = 200 nM T31543 CN3BH5 155527998 IC50 = 1258.93 nM T31543 C7SB9X 155528083 Ki = 25 nM T31543 CHYW65 155528639 IC50 = 15848.93 nM T31543 CG68UH 155529134 IC50 = 810 nM T31543 CN0B2S 155529433 Ki = 106 nM T31543 C5QT3D 155529505 Ki = 294 nM T31543 CD7O2G 155530095 IC50 = 63095.73 nM T31543 CA82SM 155530516 Ki = 2.5 nM T31543 C46AZL 155530642 Ki > 25000 nM T31543 C35QWO 155531023 IC50 = 1995.26 nM T31543 CDT7A9 155531797 IC50 > 10000 nM T31543 CER1Z8 155532768 Ki = 7.2 nM T31543 C1HAW5 155533558 IC50 = 20 nM T31543 CEFK81 155534191 Ki = 0.22 nM T31543 C7M2UT 155534310 IC50 = 30 nM T31543 C2YB0P 155535378 Ki = 4.9 nM T31543 C6AE0I 155535379 Ki = 18 nM T31543 CUV1I4 155535874 IC50 = 10000 nM T31543 C12HON 155536142 IC50 = 31622.78 nM T31543 CY6DK3 155540964 IC50 = 12.59 nM T31543 C4P2GV 155543617 Ki > 25000 nM T31543 CT4S3M 155544624 IC50 = 2100 nM T31543 C5FZ3I 155545003 Ki = 294 nM T31543 CA08GE 155545013 Ki = 188 nM T31543 CQ51DI 155546002 IC50 = 70 nM T31543 C5MB9R 155547962 IC50 = 7943.28 nM T31543 CLFB25 155548371 IC50 = 25118.86 nM T31543 CK0E7M 155548720 IC50 = 4500 nM T31543 C3R9TO 155551160 IC50 = 2400 nM T31543 CU9FL4 155551858 Ki > 50000 nM T31543 COM52R 155551892 IC50 = 10000 nM T31543 CJ3FI5 155553630 IC50 = 25118.86 nM T31543 CU8LR3 155555208 Ki > 25000 nM T31543 CM3X6Y 155555703 Ki = 11 nM T31543 CXYR84 155556203 Ki = 5.4 nM T31543 CM63SG 155557605 IC50 = 7500 nM T31543 CSW48V 155557718 IC50 = 1258.93 nM T31543 C0IW5Z 155557962 IC50 > 20000 nM T31543 C3VJ5W 155559076 Ki = 0.36 nM T31543 CY60RV 155559158 Ki = 253 nM T31543 CQ3MJ4 155559840 Ki = 3.9 nM T31543 C0B3ID 155562970 Ki = 0.5 nM T31543 C6N0LM 155564043 IC50 > 10000 nM T31543 CM8XB1 155565537 IC50 = 6309.57 nM T31543 CTF0S7 155566456 Ki = 1.3 nM T31543 CP4F1U 155567613 Ki = 480000 nM T31543 D00LOL 970375 IC50 = 570 nM T31543 D01TWD 126363 Ki = 14000 nM T31543 D07SFI 2332 Ki = 400000 nM T31543 D07ZRG 46899577 Ki = 55 nM T31543 D08KCA 72429 Ki = 696 nM T31543 D0SP2I 6852210 Ki = 46 nM T31543 D0W2SV 70689167 Ki = 0.011 nM T17140 D01BYB 5957 EC50 = 340 nM T17140 D07BSQ 5994 IC50 = 1600 nM T17140 D0H2UB 5361 EC50 = 3000 nM T17140 D0PL3N 24764487 IC50 = 45 nM T17140 D0UF2N 21706 EC50 = 500 nM T17140 CCJ8P0 440317 EC50 = 690 nM T17140 CIWV85 746996 IC50 = 7980 nM T17140 CMUV80 766793 IC50 = 14200 nM T17140 CEBX03 779113 IC50 = 29800 nM T17140 CGJ9S2 921624 IC50 = 28000 nM T17140 CYV85L 2320735 IC50 > 10000 nM T17140 CI76GD 3119320 IC50 = 4790 nM T17140 CJEV94 5287422 EC50 = 0.9 nM T17140 CDON91 5310949 EC50 = 350 nM T17140 C97WCE 5310950 EC50 = 17 nM T17140 C6P7VU 5311303 EC50 = 13000 nM T17140 CQC5W8 5702690 IC50 = 1000 nM T17140 CXUA54 5796006 IC50 = 20 nM T17140 CLF3B8 5861195 IC50 = 130 nM T17140 CLU4D6 5891789 IC50 > 10000 nM T17140 CD67GR 5897666 IC50 = 30 nM T17140 CMB71S 5922935 IC50 > 10000 nM T17140 CBA53G 5935441 IC50 = 370 nM T17140 CT5V6E 5935932 IC50 = 130 nM T17140 CDG68S 5936815 IC50 = 20 nM T17140 CX92YW 6093160 IC50 = 28500 nM T17140 CQ7U2M 6298699 IC50 = 90 nM T17140 CGAX04 6436223 IC50 = 755 nM T17140 CX7J8F 11636756 IC50 = 354.81 nM T17140 CR8U0Y 11663667 IC50 > 100000 nM T17140 C6J8WC 16066783 IC50 = 1580 nM T17140 CSXO69 16680454 IC50 = 86.1 nM T17140 C6AR3Q 16757019 IC50 = 353 nM T17140 CP0NB8 25060060 IC50 = 10 nM T17140 CG91NW 25097210 IC50 = 10 nM T17140 CG2Z1N 25097457 IC50 = 140 nM T17140 C5UOK2 25097734 IC50 = 260 nM T17140 C6ETK1 25117612 IC50 = 618 nM T17140 CJ7HT2 25117615 IC50 = 398 nM T17140 CGR1W4 25117983 IC50 = 5689 nM T17140 C8BZ0T 25117985 IC50 = 4214 nM T17140 CK06LQ 25118337 IC50 = 64 nM T17140 CQE1C2 25118338 IC50 = 69 nM T17140 C98MNR 25120809 IC50 = 441 nM T17140 CT06WO 25121155 IC50 = 2057 nM T17140 C3OC1Y 25121511 IC50 = 1271 nM T17140 CMCH17 25121856 IC50 = 613 nM T17140 CM7WO3 25122581 IC50 = 20 nM T17140 CA25BL 42603033 IC50 = 18 nM T17140 CI60EN 42666540 IC50 = 810 nM T17140 CWK71B 42795648 IC50 = 1300 nM T17140 CE25GL 42795663 IC50 = 7500 nM T17140 CQ46IG 44353592 EC50 = 80 nM T17140 CBPD97 46175179 IC50 = 398.11 nM T17140 C2W8ID 46832336 IC50 > 10000 nM T17140 C50QVP 53262865 IC50 = 438 nM T17140 C1UV0E 54590854 IC50 = 797 nM T17140 C9B6DZ 54590935 IC50 = 460 nM T17140 C2HZW4 54590936 IC50 = 920 nM T17140 CX4R5G 54590937 IC50 = 458 nM T17140 CZ41CM 54591029 IC50 = 824 nM T17140 C0Y5CL 54591030 IC50 = 1250 nM T17140 CM3T2V 57431767 IC50 = 2523 nM T17140 CE85TF 57431769 IC50 = 262 nM T17140 C8LVD4 57431775 IC50 = 324 nM T17140 C7AO1Q 57431779 IC50 = 1665 nM T17140 CS2ID6 57431780 IC50 = 1311 nM T17140 CWA65N 57431796 IC50 = 268 nM T17140 C94OEW 57431799 IC50 = 1360 nM T17140 CP4HN8 57431802 IC50 = 440 nM T17140 C06QYE 57431806 IC50 = 327 nM T17140 CVF9A8 57431849 IC50 = 67 nM T17140 CI4V2N 57431852 IC50 = 24 nM T17140 C0MBP3 57431914 IC50 = 24 nM T17140 CZTG87 57480939 IC50 = 255 nM T17140 C9ZMQ1 57480972 IC50 = 22 nM T17140 CKF4N7 57500055 IC50 = 13950 nM T17140 CBRF16 57500058 IC50 > 30000 nM T17140 CSD0M2 57658880 IC50 = 38 nM T17140 C81GJB 57658902 IC50 = 521 nM T17140 CGIP34 57658907 IC50 = 21 nM T17140 CA9WJ6 57658920 IC50 = 1947 nM T17140 CIFW58 57658935 IC50 = 115 nM T17140 C1B9DW 57658971 IC50 = 212 nM T17140 CBG3O4 58044900 IC50 = 11 nM T17140 C25PHF 58044933 IC50 > 10000 nM T17140 C2TAY8 58045034 IC50 = 203 nM T17140 CIZ69B 58045105 IC50 = 44 nM T17140 CN4Q7D 58045231 IC50 = 52 nM T17140 CG2ZR3 58045273 IC50 > 10000 nM T17140 CW5G9P 58045279 IC50 = 1020 nM T17140 CMXC37 58365250 IC50 = 16 nM T17140 C4EPA5 58365345 IC50 = 16 nM T17140 CO53TZ 58365501 IC50 = 15 nM T17140 CXY58G 58365527 IC50 = 13 nM T17140 CON6K1 58365686 IC50 = 16 nM T17140 CVP17Q 58365704 IC50 = 74 nM T17140 CB72VP 58365714 IC50 = 49 nM T17140 CZ6X0Y 58365744 IC50 = 73 nM T17140 CX8Y6Z 58365813 IC50 = 11 nM T17140 C3WB9I 58365828 IC50 = 16 nM T17140 C5CRB1 58365867 IC50 = 13 nM T17140 CF6A8Y 58365941 IC50 = 1089 nM T17140 C35RYZ 58365945 IC50 = 82 nM T17140 CJI25C 58365995 IC50 = 13 nM T17140 C3QI6Y 58366053 IC50 = 35 nM T17140 C6AC9L 58366064 IC50 = 999 nM T17140 CC67BX 58366073 IC50 = 700 nM T17140 CQAG37 59447778 IC50 = 553 nM T17140 CO7PZ5 60168729 IC50 = 10000 nM T17140 C32ADF 66895517 IC50 = 24 nM T17140 CH9Q0R 71450180 IC50 > 10000 nM T17140 CR64QG 71457337 IC50 > 10000 nM T17140 CR1L5W 71459185 IC50 = 429 nM T17140 CSV43Z 71459189 IC50 >= 10000 nM T17140 C0Y1JN 71462707 IC50 > 10000 nM T17140 C3U1YM 73669299 IC50 = 7180 nM T17140 CJYH20 76309929 IC50 = 587 nM T17140 CR93FA 76309930 IC50 = 723 nM T17140 CYQ01L 76313648 IC50 = 3300 nM T17140 C82PEC 76317151 IC50 = 145 nM T17140 CF1KS0 76320868 IC50 = 60 nM T17140 CD30RO 76324525 IC50 = 2930 nM T17140 CYPC45 76324526 IC50 = 928 nM T17140 CG5RF9 76324527 IC50 = 377 nM T17140 C4U3DT 76324528 IC50 = 652 nM T17140 CB69EX 76324694 IC50 = 15200 nM T17140 C43VZB 76328091 IC50 = 474 nM T17140 CB2G0F 76331762 IC50 = 636 nM T17140 CJN18X 76331763 IC50 = 366 nM T17140 CJ63YT 76331764 IC50 = 638 nM T17140 C71DLU 76331765 IC50 = 856 nM T17140 CMH31Y 76335353 IC50 = 1050 nM T17140 CHX09Y 108679493 IC50 = 360 nM T17140 CVQU96 118733194 IC50 = 600 nM T17140 CPO7N5 124125214 IC50 = 8300 nM T17140 CDX97M 134691714 IC50 = 840 nM T17140 CUSH91 135431092 IC50 = 2800 nM T17140 C50GNB 136082632 IC50 = 79.8 nM T17140 CQHU28 136088910 IC50 = 106 nM T17140 CO23GR 142737932 IC50 = 910 nM T17140 C3ZOV5 142737950 IC50 = 2660 nM T17140 CI7P6A 142737955 IC50 = 800 nM T17140 C4M3FP 145952869 IC50 = 21 nM T17140 C3P0KM 145953319 IC50 = 9800 nM T17140 C5IMK3 145953533 IC50 = 100 nM T17140 C8S1NH 145953535 IC50 = 3930 nM T17140 CKT0E1 145953538 IC50 = 19 nM T17140 CQ2GB7 145953759 IC50 = 72 nM T17140 CR95YQ 145954711 IC50 = 9 nM T17140 CLFO06 145954942 IC50 = 1370 nM T17140 CKMB59 145954945 IC50 = 4240 nM T17140 C8FJE9 145956116 IC50 = 560 nM T17140 CJ5XS2 145959607 IC50 = 3000 nM T17140 C3Q1DO 145960696 IC50 > 10000 nM T17140 CLS0X7 145960885 IC50 = 25 nM T17140 C9JQ8N 145961138 IC50 = 140 nM T17140 CT7UF3 145961319 IC50 > 10000 nM T17140 CC62FN 145962500 IC50 > 10000 nM T17140 CIP21K 145963223 IC50 = 5920 nM T17140 CK4R6B 145963480 IC50 = 135 nM T17140 CSF84N 145963490 IC50 = 3280 nM T17140 CEB6C4 145963681 IC50 = 10 nM T17140 CMO5J6 155511397 IC50 = 130 nM T17140 C75XNF 155511587 IC50 = 6300 nM T17140 C4J6BF 155512768 IC50 = 60 nM T17140 CB9XT1 155513864 IC50 = 15 nM T17140 CPE58H 155514125 IC50 = 8 nM T17140 CF6LV4 155514310 IC50 > 100000 nM T17140 C4JZB6 155514547 IC50 = 40 nM T17140 CM39YO 155514691 IC50 = 140 nM T17140 C7W9LA 155514822 IC50 = 85 nM T17140 CVK82Z 155514869 IC50 = 7500 nM T17140 CM3H9Q 155514887 IC50 = 8700 nM T17140 CKVY03 155515950 IC50 = 35 nM T17140 CRY41S 155517023 IC50 = 40 nM T17140 C6GCH5 155517065 IC50 = 3000 nM T17140 CLMW53 155518757 IC50 = 9900 nM T17140 C0BRX7 155519441 IC50 = 1400 nM T17140 C9HK4E 155519617 IC50 > 10000 nM T17140 CT7W8K 155519826 IC50 = 20 nM T17140 CG6JE1 155520066 IC50 = 380 nM T17140 C4LH3M 155520244 IC50 = 25 nM T17140 CT01XB 155521633 IC50 = 180 nM T17140 CY1IU5 155521709 IC50 = 35 nM T17140 CP58CD 155523291 IC50 = 180 nM T17140 CZD97E 155524156 IC50 = 440 nM T17140 CJ58QP 155524530 IC50 = 5 nM T17140 C2NWE8 155525058 IC50 = 900 nM T17140 C8R4GF 155525867 IC50 = 45 nM T17140 CM9CW2 155526224 IC50 = 5830 nM T17140 CDJ31N 155526369 IC50 = 7500 nM T17140 CU2I4R 155526703 IC50 = 20 nM T17140 C3B6EX 155526972 IC50 = 590 nM T17140 C2CQI3 155527693 IC50 = 2400 nM T17140 CL4RC9 155528080 IC50 > 2000 nM T17140 C9EL4D 155528131 IC50 = 50 nM T17140 C1NOD4 155529242 IC50 = 4110 nM T17140 CL4NQ9 155529657 IC50 = 650 nM T17140 CX12AU 155529713 IC50 = 611 nM T17140 C5BC9V 155529971 IC50 = 17500 nM T17140 C3LU9N 155530055 IC50 = 6 nM T17140 CXGC97 155530178 IC50 = 7400 nM T17140 CQX4F0 155530320 IC50 = 668 nM T17140 CKY09W 155531083 IC50 = 580 nM T17140 CYQ84G 155532585 IC50 = 10700 nM T17140 CBD9L6 155533139 IC50 = 19 nM T17140 C8QR1E 155534154 IC50 = 5000 nM T17140 C7GZ8C 155534904 IC50 = 2100 nM T17140 CJB82P 155535066 IC50 = 1310 nM T17140 CP97ML 155535352 IC50 = 65 nM T17140 CH47QU 155535354 IC50 = 390 nM T17140 C4L0SX 155537072 IC50 = 20 nM T17140 CTG39Y 155537553 IC50 = 1500 nM T17140 COQC96 155537975 IC50 = 95 nM T17140 CH9Y0J 155538262 IC50 = 10 nM T17140 CA26YF 155538734 IC50 = 11200 nM T17140 CH92GY 155539221 IC50 = 65 nM T17140 CHI78B 155540008 IC50 = 40 nM T17140 C45GAY 155540285 IC50 = 720 nM T17140 C4ZAM2 155540414 IC50 = 400 nM T17140 C9BGA0 155540772 IC50 = 700 nM T17140 C0K9FV 155542440 IC50 = 3700 nM T17140 C5OIQ7 155542766 IC50 = 7 nM T17140 COD7Q8 155543044 IC50 = 883 nM T17140 C0I3WD 155543378 IC50 = 170 nM T17140 C5AFJ7 155543528 IC50 = 850 nM T17140 CI0E4P 155544725 IC50 = 6800 nM T17140 C6L2JE 155544746 IC50 = 140 nM T17140 CCB2O4 155545366 IC50 = 7500 nM T17140 C2CZ7O 155545879 IC50 = 10000 nM T17140 CR5D3Q 155548909 IC50 = 5700 nM T17140 CS57LN 155549377 IC50 > 10000 nM T17140 C1MYS0 155549544 IC50 = 40 nM T17140 CET18Q 155550268 IC50 = 21 nM T17140 CC7AN2 155550493 IC50 = 1300 nM T17140 CSQ05B 155551563 IC50 = 15 nM T17140 CI9B5Y 155551797 IC50 = 640 nM T17140 CTBK15 155552357 IC50 = 33 nM T17140 CDH06Y 155552819 IC50 = 15 nM T17140 C0F6RT 155553704 IC50 = 48 nM T17140 C3I7BT 155553879 IC50 = 190 nM T17140 CPV2E3 155554392 IC50 = 1600 nM T17140 CJ07RZ 155554473 IC50 = 80 nM T17140 CQH57Z 155555213 IC50 = 7300 nM T17140 C09SOB 155557542 IC50 = 1400 nM T17140 CPO1H2 155557786 IC50 = 150 nM T17140 C2NBD5 155558024 IC50 = 280 nM T17140 CB5Y7A 155558453 IC50 = 1000 nM T17140 C2WFY3 155558639 IC50 = 3700 nM T17140 CZ9G8K 155559078 IC50 > 100000 nM T17140 C47VBE 155559341 IC50 = 55 nM T17140 CJCO90 155560573 IC50 = 140 nM T17140 C0PYX1 155562454 IC50 >= 100000 nM T17140 CDQ97I 155562606 IC50 = 1300 nM T17140 COL84V 155563568 IC50 = 65 nM T17140 CPM6Y0 155564816 IC50 = 1000 nM T17140 C9T5VU 155564839 IC50 = 45 nM T17140 C0AK8B 155565293 IC50 = 660 nM T17140 CJTV86 155566512 IC50 = 15 nM T17140 CVT0H6 155567668 IC50 = 3800 nM T17140 C4QDL9 155568671 IC50 = 3300 nM T17140 C9TRF0 155568988 IC50 = 750 nM T17140 CQA3R5 155569370 IC50 = 648 nM T17140 D00QLM 91557 EC50 = 740 nM T17140 D03EEO 3960826 IC50 = 58300 nM T17140 D05BFC 3978952 IC50 = 96.2 nM T17140 D05NWF 6022 EC50 > 100000 nM T17140 D05RRF 17756317 IC50 = 82.4 nM T17140 D07QYU 4881 EC50 = 240 nM T17140 D0B1KT 15953802 IC50 = 20 nM T17140 D0FF6S 16038374 IC50 > 10000 nM T17140 D0M8HU 25054651 IC50 = 32.4 nM T17140 D0U1OJ 5310983 EC50 = 350 nM T17140 D0UG4S 91532 EC50 = 9200 nM T17140 D0V4GQ 5310996 EC50 = 8800 nM T17140 D0Z0QD 3081832 IC50 = 0.0083 nM T17140 D0Z1DQ 9829395 IC50 = 35 nM T17140 D0Z6UE 25054398 IC50 = 14.3 nM T58589 D06BHG 11953367 Ki = 0.3 nM T58589 D0LI1C 44469321 IC50 > 30000 nM T58589 D0X0BI 439201 Ki > 10 nM T58589 C1ZTN0 2818985 IC50 = 3200 nM T58589 C93QUY 3102216 Ki = 500 nM T58589 C0TV9U 4227718 Ki = 45 nM T58589 C73ZFI 9804704 IC50 = 86 nM T58589 CO36FU 9852117 Ki = 5.6 nM T58589 CWL4Q7 9894973 Ki = 0.59 nM T58589 CU15TR 9897921 Ki < 10000 nM T58589 CM45KH 9919335 Ki = 24.1 nM T58589 CQ39DL 9961595 Ki = 10 nM T58589 CCP49I 9988753 Ki < 10000 nM T58589 CJ37QY 10001334 Ki = 390 nM T58589 C0X3IQ 10008626 Ki <= 5.5 nM T58589 C7YH1R 10010104 Ki <= 5.5 nM T58589 C7JE8F 10010669 Ki <= 5.5 nM T58589 C9QZ6G 10031511 Ki = 0.59 nM T58589 CGI57Y 10032895 Ki < 10000 nM T58589 CNQL86 10055774 Ki <= 5.5 nM T58589 CSYU04 10056816 Ki <= 5.5 nM T58589 C68GEM 10079793 Ki < 10000 nM T58589 CIXU90 10079797 Ki < 10000 nM T58589 CU39IK 10101294 Ki <= 5.5 nM T58589 CF4WK8 10102296 Ki < 10000 nM T58589 CXF5K1 10102599 Ki <= 5.5 nM T58589 CY8R9E 10102701 Ki < 10000 nM T58589 CNY18T 10120979 Ki = 97.5 nM T58589 CZY3I5 10128103 Ki = 2.05 nM T58589 C8POE9 10128412 Ki = 1.39 nM T58589 C27URE 10151875 Ki = 0.57 nM T58589 C4U6AG 10166801 Ki = 141 nM T58589 C0W2IY 10168110 Ki = 100 nM T58589 C3RTP5 10173772 Ki = 0.4 nM T58589 CC6M9P 10187167 Ki = 78 nM T58589 C05VWM 10187347 Ki = 28 nM T58589 CH16RG 10196170 Ki = 0.68 nM T58589 CN9G3L 10217706 Ki = 0.51 nM T58589 C7FAN6 10233880 Ki = 1.5 nM T58589 CLB35I 10239095 Ki = 0.6 nM T58589 C4OVQ0 10260476 Ki <= 5.5 nM T58589 CJ9G2K 10282203 Ki = 55 nM T58589 C01IRZ 10288906 Ki = 0.13 nM T58589 CX5CV4 10300688 Ki > 10000 nM T58589 CC87GI 10311064 Ki = 22 nM T58589 CJ1W6X 10349694 Ki <= 5.5 nM T58589 C8EP5X 10350966 Ki < 10000 nM T58589 C1TQ7U 10373970 Ki < 10000 nM T58589 CXS0E7 10388673 Ki = 11.8 nM T58589 CP14YR 10396101 Ki < 10000 nM T58589 CUS3Q8 10418252 Ki <= 5.5 nM T58589 C7X2OY 10418495 Ki <= 5.5 nM T58589 CMNA43 10418701 Ki < 10000 nM T58589 CXP97A 10439868 Ki <= 5.5 nM T58589 C90DQN 10441167 Ki < 10000 nM T58589 CX79PI 10441194 Ki < 10000 nM T58589 C49PQN 10441297 Ki < 10000 nM T58589 CLEX38 10456579 Ki = 40 nM T58589 C45PFV 10463758 Ki <= 5.5 nM T58589 CWHI15 10463818 Ki <= 5.5 nM T58589 C3ZU0G 10463883 Ki < 10000 nM T58589 C4TV3E 10875606 Ki = 1023 nM T58589 CC7VZ4 10940858 Ki > 10000 nM T58589 C2OCH6 11017305 Ki = 1.33 nM T58589 CL31CX 11039234 Ki = 13.4 nM T58589 CE26TD 11050306 Ki = 1.37 nM T58589 CNJZ59 11071992 Ki = 5.73 nM T58589 CB8PH3 11167607 Ki = 0.8 nM T58589 C6VDM5 11168954 Ki = 0.41 nM T58589 C67ZQB 11180561 Ki = 0.07 nM T58589 C3CD4H 11180748 Ki = 250 nM T58589 C84IRP 11203826 IC50 = 16 nM T58589 CR9V6S 11204003 IC50 = 11 nM T58589 CW3QO7 11213709 IC50 = 1700 nM T58589 CB31LO 11214151 Ki = 10 nM T58589 C04LNE 11214480 IC50 = 0.075 nM T58589 CK8R5Q 11214819 Ki = 0.3 nM T58589 CEWC14 11214998 IC50 = 110 nM T58589 CKA87Y 11215189 IC50 = 13 nM T58589 C3UPQ2 11215488 Ki = 0.15 nM T58589 C9NT7H 11215677 Ki = 0.1 nM T58589 CP0DT6 11215913 Ki = 1.3 nM T58589 C8VN1E 11224694 Ki = 120 nM T58589 C0N5LC 11225601 Ki = 0.5 nM T58589 CQ04GL 11227059 Ki = 3.73 nM T58589 CWON94 11238372 IC50 = 54 nM T58589 C5S9IC 11259064 Ki = 2 nM T58589 CINP41 11259614 IC50 = 82 nM T58589 CE21NL 11260745 Ki = 4.5 nM T58589 CJ2BZ3 11272685 IC50 = 1.2 nM T58589 C8R1KF 11281533 Ki = 0.83 nM T58589 CC09KZ 11283865 Ki = 0.4 nM T58589 CTJW92 11284303 Ki = 3000 nM T58589 CY1EC9 11284304 IC50 = 1.46 nM T58589 C2TW3L 11284458 Ki = 23 nM T58589 C3DQ7P 11284564 Ki = 0.5 nM T58589 CUQF93 11293092 Ki = 13 nM T58589 C2K4CM 11306090 Ki = 1.1 nM T58589 CHD87N 11307467 Ki = 1.4 nM T58589 CH4V5L 11307733 IC50 = 59 nM T58589 CG7BW3 11317669 IC50 = 16 nM T58589 CS5EH9 11319515 Ki = 0.02 nM T58589 CE4A7D 11320189 Ki = 1 nM T58589 C2J1GL 11326315 IC50 = 700 nM T58589 C41ZHJ 11330286 IC50 = 48 nM T58589 CVEZ45 11331054 Ki = 3.3 nM T58589 CE2N5Z 11340940 Ki = 1.6 nM T58589 CH2NA9 11341448 Ki = 3.8 nM T58589 C9QE3H 11341479 Ki = 0.29 nM T58589 C7IL8N 11342079 IC50 = 183 nM T58589 CGSA32 11342350 Ki = 0.46 nM T58589 CUR5A1 11342704 Ki = 0.1 nM T58589 CGU5O9 11352746 Ki = 0.2 nM T58589 CHS08F 11363856 Ki = 0.5 nM T58589 C4UXC1 11364466 IC50 = 0.48 nM T58589 CJ8LZ5 11365433 Ki = 0.07 nM T58589 CTZ8E1 11373520 IC50 = 560 nM T58589 CN95TV 11375297 Ki = 73 nM T58589 C21NFQ 11376509 Ki = 230 nM T58589 C31XME 11377529 Ki = 10 nM T58589 C2U7SZ 11386138 Ki = 0.7 nM T58589 CKB2E6 11387387 IC50 = 0.2 nM T58589 CBQ4G7 11387624 Ki = 0.2 nM T58589 CFN4Q3 11387915 Ki = 0.7 nM T58589 CPV9F1 11398971 Ki = 1.9 nM T58589 COS6U4 11399429 Ki > 1000 nM T58589 C8RH5J 11405561 IC50 = 2000 nM T58589 CUQ4X8 11420875 IC50 = 130 nM T58589 CW3R8K 11421944 Ki = 17.9 nM T58589 CF41TX 11422305 Ki = 140 nM T58589 CV68QE 11433587 Ki = 3.5 nM T58589 CI15ME 11442712 IC50 = 0.25 nM T58589 C2V5ED 11444165 IC50 = 22 nM T58589 CM03JU 11444270 IC50 = 14 nM T58589 CBIY13 11444668 Ki = 1.1 nM T58589 CFG04P 11444808 Ki = 0.01 nM T58589 CY9KC3 11452874 Ki = 200 nM T58589 CGV08Y 11454567 Ki = 30 nM T58589 C89TLC 11456015 Ki = 2.6 nM T58589 C4XW1I 11466010 Ki = 6 nM T58589 C6DGB7 11467345 Ki = 31 nM T58589 CGS0Y9 11476944 Ki = 106 nM T58589 C2DX7T 11477390 Ki = 0.7 nM T58589 C0ER8C 11478613 IC50 = 21 nM T58589 C8M0XU 11478717 IC50 = 5.2 nM T58589 C03DKV 11479448 Ki = 10 nM T58589 CUC91I 11488817 Ki = 0.7 nM T58589 C4RKM5 11495796 Ki = 3450 nM T58589 C13DVN 11498691 Ki <= 5.5 nM T58589 C4BD2X 11498853 Ki < 10000 nM T58589 CNT5H8 11505970 Ki <= 5.5 nM T58589 C5SPA8 11506007 Ki <= 5.5 nM T58589 CGH4A1 11512379 IC50 = 150 nM T58589 CO7HB4 11513104 Ki <= 5.5 nM T58589 C5M2QO 11513163 Ki <= 5.5 nM T58589 CVL4R2 11513471 Ki <= 5.5 nM T58589 CZ1QS6 11519239 Ki = 19.1 nM T58589 C8QW9F 11526655 Ki = 6.4 nM T58589 C4AZO9 11526891 Ki = 16.9 nM T58589 CV97KH 11527838 Ki <= 5.5 nM T58589 C4QK9A 11527892 Ki <= 5.5 nM T58589 CR14MO 11527906 Ki <= 5.5 nM T58589 CF37AZ 11542210 Ki <= 5.5 nM T58589 CWLX79 11546560 Ki = 63 nM T58589 C4B8LI 11549335 Ki <= 5.5 nM T58589 CMIS36 11549560 Ki <= 5.5 nM T58589 CU95QM 11549562 Ki <= 5.5 nM T58589 CR5V6E 11553268 Ki = 52000 nM T58589 C0SDP6 11555433 IC50 = 39.2 nM T58589 CD02NX 11555599 IC50 = 79 nM T58589 C2Z4WP 11561240 IC50 = 3.3 nM T58589 CU7CR4 11570120 Ki = 0.045 nM T58589 CUDQ72 11571204 Ki <= 5.5 nM T58589 C3ZQ1H 11575578 Ki = 25.5 nM T58589 CCF8U0 11577748 Ki <= 5.5 nM T58589 CD7TL4 11584184 IC50 = 84.2 nM T58589 C5JY3H 11585604 Ki <= 5.5 nM T58589 C7KN1L 11585627 Ki <= 5.5 nM T58589 CG0Q6N 11589876 Ki > 50000 nM T58589 C7XDG2 11592927 Ki <= 5.5 nM T58589 C9D7LB 11596635 Ki = 478 nM T58589 CL9M5H 11600186 Ki <= 5.5 nM T58589 CF5YX0 11600235 Ki <= 5.5 nM T58589 C90SJN 11600324 Ki < 10000 nM T58589 CW28IT 11604201 Ki = 1580 nM T58589 CCPQ75 11605512 Ki = 565 nM T58589 C1D2NQ 11614670 Ki <= 5.5 nM T58589 CXV40U 11620238 Ki = 1.8 nM T58589 C34GHD 11620871 Ki = 0.045 nM T58589 CJ06QY 11620980 Ki = 43.8 nM T58589 CRW92U 11621618 Ki <= 5.5 nM T58589 C0XZ1G 11621850 Ki <= 5.5 nM T58589 CXU7G5 11635364 IC50 = 44.9 nM T58589 CG07XP 11635365 Ki = 4.1 nM T58589 CJAD90 11636064 Ki <= 5.5 nM T58589 CC0P7Y 11636119 Ki <= 5.5 nM T58589 CPR35B 11636121 Ki <= 5.5 nM T58589 CL7N1Z 11641218 Ki = 462 nM T58589 C5PZ3J 11650337 Ki <= 5.5 nM T58589 CFB32S 11650783 Ki <= 5.5 nM T58589 C9DON1 11657717 Ki <= 5.5 nM T58589 CQXI09 11663606 Ki = 41.4 nM T58589 C9ESF1 11663809 Ki = 1.7 nM T58589 C42RFY 11670114 Ki = 752 nM T58589 C82AWM 11670860 Ki = 23.5 nM T58589 CO5R3C 11671905 Ki <= 5.5 nM T58589 CFA5K1 11672186 Ki <= 5.5 nM T58589 C65VUE 11672243 Ki <= 5.5 nM T58589 C7QCH6 11676747 Ki = 1645 nM T58589 C06SLD 11679144 Ki <= 5.5 nM T58589 CKF81H 11685446 IC50 = 9.9 nM T58589 C5QC8X 11686256 Ki <= 5.5 nM T58589 C1R7VL 11686399 Ki <= 5.5 nM T58589 C2BTI0 11691896 Ki = 59.9 nM T58589 C8Y4US 11699718 Ki <= 5.5 nM T58589 CZB59C 11707335 Ki <= 5.5 nM T58589 C4PY9R 11707423 Ki <= 5.5 nM T58589 C4CA1S 11707528 Ki <= 5.5 nM T58589 CYG71V 11714620 Ki <= 5.5 nM T58589 C28ZVE 11719314 Ki = 119 nM T58589 CH9P6I 11752335 Ki = 9.5 nM T58589 C8Q6ZV 11757682 Ki = 0.02 nM T58589 C3NI6Q 11766718 Ki < 10000 nM T58589 C31JUX 11786597 Ki = 1.09 nM T58589 C9LRU7 11848206 Ki = 0.26 nM T58589 C4MQ2U 12085129 Ki = 65 nM T58589 CI2Z4V 12085130 Ki = 15 nM T58589 CI72ED 12085131 Ki = 12 nM T58589 CK6OS9 12085225 Ki = 63.5 nM T58589 CC76XK 12085227 Ki = 85 nM T58589 C1V9EY 16041612 Ki = 0.2 nM T58589 CNFS70 16047262 Ki = 4.4 nM T58589 C48JMD 16102881 Ki = 2.95 nM T58589 CCHB78 16102882 Ki = 13.5 nM T58589 C6EJP9 16102883 Ki = 0.54 nM T58589 C03DLN 16102884 Ki = 2.5 nM T58589 CAQ93H 16102885 Ki = 2.8 nM T58589 CYS6P1 16102896 Ki = 0.81 nM T58589 C2DI6U 16102897 Ki = 0.44 nM T58589 CQT8E1 16102898 Ki = 0.66 nM T58589 CF89EI 16102899 Ki = 1.44 nM T58589 CYN40W 16102907 Ki = 1.47 nM T58589 CXZ5J9 16102908 Ki = 11.6 nM T58589 C68KPL 16102909 Ki = 119 nM T58589 CO7L1Z 16102918 Ki = 0.93 nM T58589 CCP79J 16102919 Ki = 10.3 nM T58589 C9GF5P 16102920 Ki = 1.35 nM T58589 CMIV80 16102922 Ki = 62.5 nM T58589 CUF20D 16102923 Ki = 1.95 nM T58589 CB43PJ 16105690 Ki < 10000 nM T58589 CC7S8Z 16105694 Ki < 10000 nM T58589 CLM34B 16105696 Ki < 10000 nM T58589 CZ8PH5 16105698 Ki < 10000 nM T58589 CXK4E7 16105701 Ki < 10000 nM T58589 CB4N2X 16105703 Ki < 10000 nM T58589 C8U2YI 16105727 Ki < 10000 nM T58589 CVI42S 16105729 Ki < 10000 nM T58589 CICB86 16105734 Ki < 10000 nM T58589 CR85GM 16105742 Ki < 10000 nM T58589 CFQ42K 16105746 Ki < 10000 nM T58589 C6LSG9 16105751 Ki < 10000 nM T58589 CL4ZQ8 16108953 IC50 <= 4000 nM T58589 CQAH63 16108958 IC50 > 4000 nM T58589 CL7R0B 16108960 Ki = 1.6 nM T58589 C12LZJ 16108962 Ki = 17 nM T58589 CNPJ98 16108963 Ki = 143 nM T58589 CKM75I 16108964 IC50 = 1700 nM T58589 CBL7U8 16108965 IC50 = 14 nM T58589 C3VC2M 16108966 Ki = 17 nM T58589 CL90BF 16108967 IC50 = 359 nM T58589 CX0BL6 16108968 Ki = 132 nM T58589 CMX85A 16108969 Ki = 0.24 nM T58589 CZ84ND 16202227 Ki = 1.2 nM T58589 C8H9YA 16220913 Ki = 308 nM T58589 CC2ZD8 16220914 Ki = 138 nM T58589 C7GX3R 16220915 Ki = 8.3 nM T58589 CA20GX 16220916 Ki = 5.4 nM T58589 CYIC03 16220917 Ki = 84.8 nM T58589 CO6KJ2 16220918 Ki = 3.7 nM T58589 C1QE6G 16220986 Ki = 393 nM T58589 CIAQ15 16220987 Ki = 27.7 nM T58589 CKJX76 16220988 Ki = 367 nM T58589 CS4U5I 16220989 Ki = 77.6 nM T58589 CV3AI0 16220990 Ki = 7.6 nM T58589 CC65FR 16221053 Ki = 25.2 nM T58589 CRP3N0 16221054 Ki = 20.6 nM T58589 CX2J9P 16221055 Ki = 4.8 nM T58589 C96BGW 16221056 Ki = 14 nM T58589 CSP6I0 16221057 Ki = 5.9 nM T58589 C04COE 16221108 Ki = 5.5 nM T58589 C3NF9J 16221109 Ki = 5 nM T58589 CK0XQ9 16221110 Ki = 8.9 nM T58589 CJG3C2 16221111 Ki = 5 nM T58589 CE83RF 16221160 Ki = 21.8 nM T58589 CG4D0Z 16221161 Ki = 5.7 nM T58589 C7QS0G 16221162 Ki = 13.4 nM T58589 C8CP4Q 16221163 Ki = 132 nM T58589 C4HP1S 16221164 Ki = 24.8 nM T58589 C2M8KF 16221225 Ki = 127 nM T58589 CMJ02P 16221226 Ki = 40.6 nM T58589 CSA49K 16221227 Ki = 120 nM T58589 CD67GW 16221228 Ki = 4.7 nM T58589 CTI5B7 16221229 Ki = 10 nM T58589 CIWM58 16221282 Ki = 0.4 nM T58589 CX2E1R 16221283 Ki = 6.7 nM T58589 C6M4LX 16726096 Ki = 0.5 nM T58589 CUG94I 16726109 Ki = 0.77 nM T58589 CX2MU3 16747694 IC50 = 0.45 nM T58589 C90IKR 17751347 IC50 = 1.53 nM T58589 CDE6M1 17751422 IC50 = 130 nM T58589 C8F4VI 17751599 IC50 = 1210 nM T58589 C0L5FH 17751827 IC50 = 25.2 nM T58589 CS8RD0 17751868 IC50 = 2040 nM T58589 CN82VK 23627396 Ki = 3.1 nM T58589 CIFA02 23627458 Ki = 4.7 nM T58589 C52ZOX 23627520 Ki = 15.5 nM T58589 C9C3UF 23627521 Ki = 1.7 nM T58589 CK8XN7 23627523 Ki = 9.1 nM T58589 CAT48V 23627583 Ki = 8.9 nM T58589 CY46XI 23628223 Ki = 0.4 nM T58589 CL45YA 23630509 IC50 = 290 nM T58589 C0LI6H 23630510 IC50 = 210 nM T58589 C86RLI 23630511 IC50 = 3.9 nM T58589 CZMB41 23630512 IC50 = 9.3 nM T58589 C0KME3 23630513 IC50 = 49 nM T58589 C8C1FO 23630514 IC50 > 10000 nM T58589 CN9MI8 23630612 IC50 = 640 nM T58589 CX8UN7 23630613 IC50 = 12 nM T58589 C30ZPG 23630614 IC50 = 71 nM T58589 CKE90S 23630615 IC50 = 1600 nM T58589 CVW34A 23630715 IC50 = 1.8 nM T58589 CQ65JF 23630809 IC50 = 60 nM T58589 C2VFP3 23630810 IC50 = 200 nM T58589 CV4SN3 23630811 IC50 = 23 nM T58589 C2TNP5 23630812 IC50 > 10000 nM T58589 CPM6B8 23630813 IC50 = 10 nM T58589 C9XQZ8 23630814 IC50 = 650 nM T58589 CR43ZH 23630918 IC50 = 44 nM T58589 C9CH0A 23630919 IC50 = 3.5 nM T58589 C9EQ7K 23630920 IC50 = 1200 nM T58589 CJ85EN 23630923 IC50 > 10000 nM T58589 CLOX15 23631015 IC50 = 320 nM T58589 CF0GB7 23631902 IC50 = 3 nM T58589 C9ZAV1 23631903 IC50 = 13 nM T58589 CET97P 24884552 Ki = 0.41 nM T58589 CRAK17 24893993 Ki = 0.7 nM T58589 CE8G9Z 24895111 Ki = 251 nM T58589 C38XVG 24895112 Ki = 65 nM T58589 C24RIT 24895113 Ki > 10000 nM T58589 CD4S1J 24895114 Ki = 108 nM T58589 CCF80B 24895181 Ki = 56 nM T58589 CT9V3Q 24895182 Ki = 28 nM T58589 C2MIR3 24895183 Ki = 72 nM T58589 CC2UH9 24895184 Ki = 24 nM T58589 C4BAU6 24895185 Ki > 10000 nM T58589 C4Z6JT 24895186 Ki = 217 nM T58589 C07VXH 24895252 Ki = 19 nM T58589 C4LQ8N 24895253 Ki = 1.2 nM T58589 CRDU93 24895255 Ki = 5.6 nM T58589 CT5GY9 24895256 Ki = 24 nM T58589 C1N0CZ 24895351 Ki = 23 nM T58589 CRQ6V5 24895352 Ki = 70 nM T58589 CZV68P 24895353 Ki = 331 nM T58589 C4GP1S 24895354 Ki = 202 nM T58589 CKN0E1 24895355 Ki = 431 nM T58589 CY9LI6 24895449 Ki = 43 nM T58589 C60SUP 24895450 Ki = 215 nM T58589 CI2S7Y 24895452 Ki = 0.25 nM T58589 CQ9N6Z 24895454 Ki = 2.1 nM T58589 C32FHS 24895455 Ki = 15 nM T58589 CU31LR 24895550 Ki = 0.6 nM T58589 CVDK89 24970287 IC50 = 0.12 nM T58589 CNIX27 24970501 Ki = 67 nM T58589 CGO65I 24970503 Ki = 1996 nM T58589 CPR90J 25181410 Ki = 11 nM T58589 C0I6QH 25181411 Ki = 93 nM T58589 CF3ZB9 25195622 Ki = 0.12 nM T58589 C79QTD 25207727 IC50 = 125 nM T58589 CQ0K9H 42605727 IC50 = 3100 nM T58589 C7B4AG 42606173 IC50 = 500 nM T58589 CKD3V8 42606292 IC50 = 5 nM T58589 CK19AE 44355038 Ki > 10000 nM T58589 C7JZ8G 44391943 Ki > 5000 nM T58589 CUA0Z6 44391956 Ki > 5000 nM T58589 CD90BO 44391962 Ki = 385 nM T58589 C91YGR 44391977 Ki = 250 nM T58589 CPAZ59 44391980 Ki = 35 nM T58589 C1O8FA 44391982 Ki > 5000 nM T58589 CB6M8N 44392010 Ki = 3500 nM T58589 CIR9X3 44392012 Ki = 130 nM T58589 C27IOC 44392025 Ki = 11 nM T58589 C1S6KP 44392040 Ki = 38 nM T58589 C2A8BO 44392045 Ki = 25 nM T58589 C0D9QZ 44392064 Ki > 5000 nM T58589 CZP3F2 44392068 Ki = 2 nM T58589 CZV49W 44392113 Ki = 730 nM T58589 CD24PS 44392133 Ki = 54 nM T58589 CGDY20 44392138 Ki = 126 nM T58589 C82CAK 44392156 Ki = 2.2 nM T58589 CN3T6R 44392544 Ki = 130 nM T58589 C3QK1W 44401703 Ki = 230 nM T58589 CN3CQ8 44401768 Ki = 1280 nM T58589 CE30XP 44401834 Ki = 33 nM T58589 CDS12U 44401887 Ki = 119 nM T58589 CW5TK9 44401932 Ki = 11 nM T58589 CI9Z8T 44402028 Ki = 11.5 nM T58589 C8H2YK 44402075 Ki = 200 nM T58589 CTW7N2 44402076 Ki = 11 nM T58589 C93VON 44402279 Ki = 88 nM T58589 CO5D1X 44402298 Ki = 6 nM T58589 CU64BX 44410020 IC50 = 1100 nM T58589 C4FD7Y 44410026 IC50 = 95 nM T58589 CM1JP7 44410059 IC50 > 40000 nM T58589 CR9WY5 44410084 IC50 = 700 nM T58589 CA7PS8 44410143 IC50 = 1700 nM T58589 CRP3X2 44410179 IC50 = 540 nM T58589 C2GR1F 44410186 IC50 = 210 nM T58589 CTP46F 44410250 IC50 = 220 nM T58589 CW8G2V 44410254 IC50 = 4300 nM T58589 C91LOM 44410269 IC50 = 590 nM T58589 C03ZNS 44410273 IC50 = 560 nM T58589 CNV1L9 44410313 IC50 = 780 nM T58589 CZQX26 44410316 IC50 = 73 nM T58589 C2B5EM 44410328 IC50 = 62 nM T58589 C3RCW8 44410368 IC50 = 960 nM T58589 C4R3HA 44410972 Ki = 2100 nM T58589 C9D6BT 44411050 Ki = 184 nM T58589 C5MEF4 44411051 Ki = 3.4 nM T58589 CI2Q5H 44411054 Ki = 1.7 nM T58589 C9EWK7 44411058 Ki = 9.5 nM T58589 C7OBM1 44411062 Ki = 1.4 nM T58589 CLM3B0 44411068 Ki = 5.2 nM T58589 CE43KC 44411071 Ki = 28 nM T58589 CD9EZ1 44411080 Ki = 26 nM T58589 CZS4U1 44411091 Ki = 70 nM T58589 C9K2LJ 44411092 Ki = 80 nM T58589 CB41DZ 44411093 Ki = 1.7 nM T58589 CQKX13 44411095 Ki = 2.2 nM T58589 C07CPD 44411101 Ki = 1.5 nM T58589 C6NC8V 44411134 Ki = 893 nM T58589 CCLW04 44411135 Ki = 9.1 nM T58589 CGRY62 44411138 Ki = 3.5 nM T58589 C31BMX 44411153 Ki = 52 nM T58589 CKU49L 44411245 Ki = 62 nM T58589 C2VKS7 44411252 Ki = 65 nM T58589 C8M6FY 44411294 Ki = 0.71 nM T58589 CQE41C 44411297 Ki = 815 nM T58589 C5H1NY 44411338 Ki = 611 nM T58589 C1EA5B 44411343 Ki = 4 nM T58589 CDY70Z 44411344 Ki > 3000 nM T58589 C23YEB 44411345 Ki > 3000 nM T58589 CQ2BI1 44411347 Ki = 25 nM T58589 C68QXN 44411349 Ki = 213 nM T58589 CE74PI 44411353 Ki = 2.9 nM T58589 CDH8E9 44411355 Ki = 17 nM T58589 CI8O0K 44411358 Ki = 1.5 nM T58589 CO31SL 44411360 Ki = 23 nM T58589 CZ6P9W 44411364 Ki = 1.5 nM T58589 CN5P0A 44411368 Ki = 3.3 nM T58589 C0G9HJ 44411372 Ki = 8 nM T58589 CGF61K 44411392 Ki = 34 nM T58589 CTW96R 44411393 Ki = 5.5 nM T58589 CN2G9R 44411442 Ki = 2.8 nM T58589 CUE29X 44411452 Ki = 0.85 nM T58589 C2W3DT 44411457 Ki = 3.4 nM T58589 CLI08P 44412007 Ki <= 5.5 nM T58589 C4KJR5 44412412 Ki <= 5.5 nM T58589 CNZG76 44418930 Ki = 0.81 nM T58589 C6MQF3 44419045 IC50 = 6.4 nM T58589 C1YPW0 44419046 IC50 = 325 nM T58589 C9KZ5O 44419100 IC50 = 540 nM T58589 C79FXT 44421279 Ki = 1.2 nM T58589 CEO74Z 44428099 IC50 > 10000 nM T58589 CP4Y3S 44428100 IC50 = 1100 nM T58589 CX5C2J 44430679 Ki = 1451 nM T58589 CM6NO2 44430680 Ki = 14 nM T58589 CGP0N8 44430681 Ki = 18 nM T58589 CY4WJ2 44430682 Ki = 3.7 nM T58589 CA8Q7N 44430683 Ki = 60 nM T58589 C0WTZ7 44430684 Ki = 24.5 nM T58589 C8OLK2 44430685 Ki = 49 nM T58589 COI8Z0 44430686 Ki = 2 nM T58589 C65ONB 44430687 Ki = 30 nM T58589 C0H1ES 44430688 Ki = 4.9 nM T58589 CBR46X 44430692 Ki = 3.7 nM T58589 C8S2ZG 44430694 Ki = 3.6 nM T58589 CRF25T 44430696 Ki = 0.4 nM T58589 C5G6TD 44432176 Ki = 134 nM T58589 CFB18H 44432178 Ki = 7.6 nM T58589 CRBX21 44432181 Ki = 1.45 nM T58589 CVN93I 44432186 Ki = 0.68 nM T58589 C49NAQ 44432198 Ki = 1.85 nM T58589 C3ZJ5F 44432207 Ki = 2.4 nM T58589 CC5TL6 44432212 Ki = 1.58 nM T58589 CYGL73 44432215 Ki = 1.1 nM T58589 C64XDP 44432220 Ki = 2.6 nM T58589 COR0T7 44432221 Ki = 1.2 nM T58589 CC47IB 44432222 Ki = 1.8 nM T58589 CGC75O 44432223 Ki = 3.8 nM T58589 CVZ18Y 44455004 Ki = 0.43 nM T58589 CZ39GO 44455035 Ki = 0.59 nM T58589 COGS39 44455038 Ki = 0.66 nM T58589 CTV8X4 44455073 Ki = 0.79 nM T58589 CEPR21 44455074 Ki = 579 nM T58589 C50PNH 44455075 Ki = 0.35 nM T58589 C0F3MC 44455087 Ki = 0.4 nM T58589 C9T0EJ 44455089 Ki = 1.5 nM T58589 C07XKW 44455090 Ki = 0.6 nM T58589 C0B1NM 44455107 Ki = 83.5 nM T58589 CY0JU1 44455108 Ki = 24.5 nM T58589 CXSR48 44455145 Ki = 88.5 nM T58589 CJ1MN2 44455147 Ki = 479 nM T58589 C9UKR8 44455148 Ki = 71.5 nM T58589 CSFA12 44455150 Ki = 109 nM T58589 CL37VJ 44455181 Ki = 660 nM T58589 C9X0BM 44455182 Ki = 1050 nM T58589 CL1Q8W 44455227 Ki = 1090 nM T58589 CNVJ71 44455228 Ki = 95 nM T58589 CDB65J 44455229 Ki = 125 nM T58589 CD9CZ7 44455255 Ki = 516 nM T58589 CXE54J 44455256 Ki = 59.1 nM T58589 CD64NE 44455268 Ki = 0.4 nM T58589 C8Q6JE 44455364 Ki = 1.2 nM T58589 C9XP0N 44455366 Ki = 1.5 nM T58589 CQ5EP2 44455492 Ki = 2.3 nM T58589 C8UBI3 44455519 Ki = 0.2 nM T58589 CT7HW2 44455549 Ki = 1.3 nM T58589 CZ1O6I 44455574 Ki = 0.9 nM T58589 C72CFO 44455853 Ki = 1.8 nM T58589 C8YF9S 44455875 Ki = 0.9 nM T58589 CP8A9I 44561641 Ki = 100 nM T58589 C4LZH6 44561643 IC50 = 4.5 nM T58589 CF0B5N 44561786 Ki = 1.5 nM T58589 CHM8G3 44569935 Ki = 21 nM T58589 CPS43A 44569936 Ki = 34 nM T58589 CN8DZ2 44569937 Ki = 113 nM T58589 C2MK9Z 44569938 Ki = 149 nM T58589 CKE5P6 44569939 Ki = 210 nM T58589 CSA47P 44569940 Ki = 410 nM T58589 C1SOB8 44570026 Ki = 1090 nM T58589 C5I0QO 44570136 Ki = 1210 nM T58589 CC36VK 44570137 Ki = 1570 nM T58589 CTRU56 44570138 Ki = 2200 nM T58589 CGD34W 44570139 Ki = 13010 nM T58589 C3C2YB 44579694 IC50 = 1.8 nM T58589 C3J1KC 44580047 Ki = 1.6 nM T58589 C5E8RX 44580048 Ki = 0.69 nM T58589 C5J1YQ 44580049 Ki = 0.67 nM T58589 C3WPQ9 44580209 Ki = 0.96 nM T58589 CNM2H1 44580742 Ki = 0.8 nM T58589 CTD24M 44580743 Ki = 0.48 nM T58589 CBLK51 44580744 Ki = 0.39 nM T58589 C0GI6R 44587041 IC50 = 1.2 nM T58589 C2PD7R 44587181 IC50 = 0.8 nM T58589 CLT2G5 44587182 IC50 = 1 nM T58589 C58RKS 44587183 Ki = 0.7 nM T58589 C90QHG 44587184 Ki = 0.44 nM T58589 CL3IJ1 44587185 Ki = 1.1 nM T58589 C7USG0 44587186 Ki = 0.15 nM T58589 CYW1F6 44587187 Ki = 0.1 nM T58589 CF0C2O 44587188 IC50 = 0.37 nM T58589 CE23AR 44587189 IC50 = 0.14 nM T58589 CC3R0G 44587206 IC50 = 62 nM T58589 C8ZOV4 44587207 IC50 = 23 nM T58589 C2BXO7 44593650 Ki = 0.67 nM T58589 CC9S4T 46216675 IC50 = 0.19 nM T58589 C8JZI3 46216744 IC50 = 4.6 nM T58589 CTU3R5 46216844 IC50 = 1.5 nM T58589 CB0I2Z 46216845 IC50 = 1.8 nM T58589 CT4D1V 46216846 IC50 = 1 nM T58589 C12HXW 46216847 IC50 = 0.6 nM T58589 C6LK7W 46229895 IC50 > 10000 nM T58589 CL4N5G 46229967 IC50 = 1.3 nM T58589 C13TMX 46229968 IC50 = 28 nM T58589 C2YNW1 46230011 IC50 > 1000 nM T58589 C9JK7D 46230012 IC50 > 1000 nM T58589 CD7ZC6 46230013 IC50 > 1000 nM T58589 CAI50D 46230067 IC50 = 1 nM T58589 C7RJH9 46230068 IC50 = 4.4 nM T58589 CWJ9F0 46230069 IC50 = 15 nM T58589 C8JA3U 46230119 IC50 = 0.43 nM T58589 CT01AD 46230120 IC50 = 0.26 nM T58589 C4M3EK 46230121 IC50 = 0.13 nM T58589 CJ41PR 46230160 IC50 = 0.2 nM T58589 CH1RE9 46230161 IC50 = 0.14 nM T58589 CX20BL 46230162 IC50 = 1.3 nM T58589 CJ6FU3 46230163 IC50 = 0.48 nM T58589 CPE7O4 46230202 IC50 = 0.64 nM T58589 CQY4E2 46230203 IC50 = 0.28 nM T58589 CW2D5A 46230258 IC50 = 180 nM T58589 C9H0CP 46230259 IC50 = 35000 nM T58589 CI9JZ4 46230306 IC50 = 42000 nM T58589 C5LB0M 46230307 IC50 = 6100 nM T58589 CLHZ96 46230308 IC50 = 3500 nM T58589 CHD4I0 46230309 IC50 = 0.7 nM T58589 C4KT1A 46230310 IC50 = 85 nM T58589 CI9K6A 46230352 IC50 = 1.7 nM T58589 C42UCQ 46230354 IC50 = 3.5 nM T58589 CUW9M7 46230403 IC50 = 1.6 nM T58589 C1A6WU 46230404 IC50 = 0.3 nM T58589 C9D3PW 46230458 IC50 = 7.7 nM T58589 C4VHS6 46230459 IC50 = 1.7 nM T58589 C2E8PK 46230833 IC50 = 1.2 nM T58589 C1H7LY 46230834 IC50 = 17 nM T58589 C06HIR 46230835 IC50 = 2.3 nM T58589 CXS6D0 46230836 IC50 = 31 nM T58589 C26ZJX 46230889 IC50 = 3.6 nM T58589 CD7CV8 46230890 IC50 = 32 nM T58589 C1LIK9 46230891 IC50 > 100 nM T58589 C2VEI6 46230892 IC50 = 59 nM T58589 CG5N0L 46230893 IC50 = 17 nM T58589 CNO24Q 46230938 IC50 = 4.6 nM T58589 CLX87C 46230939 IC50 = 1 nM T58589 CA34LI 46230940 IC50 = 1.4 nM T58589 CGK92B 46230941 IC50 = 0.8 nM T58589 C98JCN 46230989 IC50 = 3.9 nM T58589 CG03LI 46230990 IC50 = 0.5 nM T58589 CK74NF 46911683 IC50 = 1.3 nM T58589 C8A5JH 46911684 Ki = 4.6 nM T58589 COWR30 49863227 Ki = 34 nM T58589 C2S4KB 49863228 Ki = 14 nM T58589 CN6CE1 49863229 Ki = 12 nM T58589 C08ENG 49863230 Ki = 12 nM T58589 CSO1T6 49863231 Ki = 78 nM T58589 CAY62R 49863232 Ki = 21 nM T58589 C42HRX 49863233 IC50 = 23 nM T58589 CGYV42 49863234 Ki = 16 nM T58589 CWI61B 49863235 Ki = 11 nM T58589 C7L9WC 49863236 Ki = 3.4 nM T58589 CU2Y0N 49863237 Ki = 30 nM T58589 C2YXJ6 53248885 Ki = 0.1 nM T58589 CQSV19 53360054 IC50 = 0.43 nM T58589 CK7F3Y 54580628 Ki = 0.17 nM T58589 CQ8C9G 54580655 Ki = 17.6 nM T58589 C3KW6G 54581634 Ki = 0.21 nM T58589 CYDG96 54581635 IC50 = 0.43 nM T58589 CN3GY5 54581664 IC50 = 3.6 nM T58589 CXZ2T7 54581665 Ki = 718 nM T58589 CZD8U9 54581666 Ki = 1.98 nM T58589 CDHJ78 54581667 Ki = 0.52 nM T58589 CAFY01 54582655 Ki = 0.11 nM T58589 CKC3G4 54582656 Ki = 1.09 nM T58589 CTRO07 54583583 IC50 = 475 nM T58589 C84KJN 54583617 Ki = 0.18 nM T58589 C9TVP7 54584600 IC50 = 2.2 nM T58589 CL92WT 54585539 Ki = 60 nM T58589 CJIV69 54585540 IC50 = 1.28 nM T58589 C4STF5 54586518 IC50 = 98.6 nM T58589 CJ04HM 54586519 Ki = 0.22 nM T58589 CDP6V3 54587514 IC50 = 0.49 nM T58589 C45WVG 54587550 Ki = 31.8 nM T58589 CCU28P 54587551 Ki = 541 nM T58589 CI38WG 54587552 Ki = 0.5 nM T58589 C0VM3Y 54587553 Ki = 1.6 nM T58589 CHA35B 54772237 IC50 = 0.09 nM T58589 CSIT41 56589598 IC50 = 0.3 nM T58589 CCGQ04 56594241 Ki = 64 nM T58589 CQK5I0 56594242 Ki = 183 nM T58589 CRBD81 56594243 Ki = 331 nM T58589 CWL18E 56594244 Ki > 10000 nM T58589 CW78HM 56594371 Ki = 159 nM T58589 C4G2SE 56594372 Ki = 18 nM T58589 C3UI1N 56594373 IC50 = 3405 nM T58589 CHUP45 56594374 Ki = 35 nM T58589 CI27CK 56594375 Ki > 10000 nM T58589 C2GJ3O 56594504 Ki = 614 nM T58589 CWXM09 56594505 Ki = 52 nM T58589 CTN0H2 56594506 Ki = 29 nM T58589 CW75EL 56594507 Ki = 214 nM T58589 CPAQ52 56594508 Ki = 98 nM T58589 C2L9SG 56594639 Ki = 418 nM T58589 CD3E4Y 56594640 Ki = 1.9 nM T58589 CNIP32 56594641 Ki = 3.5 nM T58589 CW1A5M 56594642 Ki = 0.9 nM T58589 C6HLO4 56594643 Ki = 198 nM T58589 C9LF2Q 56594768 Ki = 4.7 nM T58589 C92MLU 56594769 IC50 = 0.18 nM T58589 CY9JD5 56594770 Ki = 3.1 nM T58589 CS76GP 56594771 Ki = 69.9 nM T58589 CVK17L 56594772 IC50 = 1.1 nM T58589 C0UW1N 56658544 Ki = 296 nM T58589 CU9NQ4 56668920 Ki = 565 nM T58589 CV80AB 56672397 IC50 = 1371 nM T58589 CJ0A1B 56679097 Ki = 311 nM T58589 CU0Z1C 56835162 Ki = 4 nM T58589 C7VM9I 56835163 IC50 = 12 nM T58589 CQO75F 56951319 IC50 = 83.9 nM T58589 CTV6P0 57342336 Ki = 2.1 nM T58589 C7O2KQ 57342494 Ki = 3.1 nM T58589 CIY7G9 57342496 Ki = 4.2 nM T58589 C5B9QU 57342845 Ki = 2.8 nM T58589 CH0Q2J 57342847 Ki = 5.5 nM T58589 CF3ET1 57342849 Ki = 4.3 nM T58589 C2N0VG 57342852 Ki = 6.8 nM T58589 C3M1OD 57343016 Ki = 142 nM T58589 CZG03B 57390218 IC50 = 0.4 nM T58589 CJI47Q 57390219 IC50 = 18.7 nM T58589 C49OBW 57390411 IC50 = 7.51 nM T58589 C7W1CO 57390466 Ki > 10000 nM T58589 C5U6AL 57390932 IC50 = 17 nM T58589 C8T5HQ 57390933 IC50 = 279 nM T58589 C14PSN 57391172 IC50 = 25.9 nM T58589 C38SYJ 57391173 IC50 = 0.28 nM T58589 CUAX92 57391276 Ki > 10000 nM T58589 CEI42Q 57391278 Ki > 10000 nM T58589 CR4CU9 57392146 Ki > 10000 nM T58589 C24BYU 57392728 IC50 = 186 nM T58589 CK65VI 57392940 IC50 = 0.42 nM T58589 CD68LS 57392941 IC50 = 0.247 nM T58589 CYDF85 57393059 Ki > 10000 nM T58589 CAC8M5 57393061 Ki > 10000 nM T58589 C2CO0A 57394682 IC50 = 990 nM T58589 CZ6KQ1 57394683 IC50 = 1.38 nM T58589 C7FR2W 57394684 IC50 = 1.09 nM T58589 CRZL24 57394685 IC50 = 1.12 nM T58589 CTB9H6 57394686 IC50 = 19 nM T58589 C9TU1X 57394687 IC50 = 38 nM T58589 CH1JC4 57394688 IC50 = 23.4 nM T58589 CD2J8Z 57394689 IC50 = 4.75 nM T58589 COG8S6 57394779 Ki > 10000 nM T58589 C8PVE2 57394782 Ki > 10000 nM T58589 C2TQ5A 57394783 Ki > 10000 nM T58589 CWYQ56 57395448 IC50 = 0.28 nM T58589 CXN8Q3 57395449 IC50 = 836 nM T58589 CDH04R 57395450 IC50 = 94.7 nM T58589 CVX7F9 57395451 IC50 = 36.1 nM T58589 CYKA40 57395702 IC50 = 40.8 nM T58589 COK0D3 57396212 Ki = 1616 nM T58589 CS58YL 57396445 IC50 = 17.7 nM T58589 C95WJK 57396446 IC50 = 0.63 nM T58589 CW5K9S 57396447 IC50 = 0.22 nM T58589 CJE35F 57396534 Ki > 10000 nM T58589 C97VSN 57396535 Ki > 10000 nM T58589 C8UG2C 57396537 Ki > 10000 nM T58589 C5FV8O 57396539 Ki > 10000 nM T58589 C7H6TJ 57397292 IC50 = 0.084 nM T58589 CK3S0J 57397547 Ki > 10000 nM T58589 C20SLV 57398013 IC50 = 799 nM T58589 CWG42N 57398235 IC50 = 0.51 nM T58589 C4FRJ1 57398236 IC50 = 0.74 nM T58589 C7GA2X 57398237 IC50 = 0.65 nM T58589 C0B9RS 57398238 IC50 = 0.28 nM T58589 C17FCZ 57398239 IC50 = 20.3 nM T58589 CM07WZ 57398323 Ki > 10000 nM T58589 CG5S2A 57398325 Ki > 10000 nM T58589 CDVK40 57398327 Ki > 10000 nM T58589 C3RS9A 57398978 IC50 = 0.21 nM T58589 CM7VX0 57398979 IC50 = 178 nM T58589 CI4H6K 57398980 IC50 = 21.6 nM T58589 CV2NF8 57399227 Ki > 10000 nM T58589 CGFP58 57399382 IC50 = 2.7 nM T58589 CC5B3W 57399670 IC50 = 7 nM T58589 CEY8B9 57399671 Ki = 15 nM T58589 CU03OI 57399885 IC50 = 314 nM T58589 C1W6YL 57399886 IC50 = 152 nM T58589 CZ61BH 57399887 IC50 = 136 nM T58589 C8VG0D 57399981 Ki > 10000 nM T58589 C5BK7O 57399982 Ki > 10000 nM T58589 CH8K5Y 57400696 IC50 = 0.23 nM T58589 CU57BH 57400697 IC50 = 72.2 nM T58589 CJ3AE0 57400937 IC50 = 96 nM T58589 C4KTX6 57400985 Ki > 10000 nM T58589 CON6W8 57401425 IC50 = 98 nM T58589 CJ5M3L 57401426 Ki = 42 nM T58589 C2R6WU 57401663 IC50 = 1.47 nM T58589 C39QYA 57401664 IC50 = 0.31 nM T58589 C05JCX 57401770 Ki > 10000 nM T58589 C1JMA0 57401772 Ki > 10000 nM T58589 C91ALU 57401773 Ki > 10000 nM T58589 CJX89L 57401775 Ki > 10000 nM T58589 CB0I3M 57401777 Ki > 10000 nM T58589 C0HP6R 57401779 Ki > 10000 nM T58589 CB4T8H 57401781 Ki > 10000 nM T58589 CB2XH5 57401783 Ki > 10000 nM T58589 CXLU20 57402467 IC50 = 8.95 nM T58589 C3C9JU 57402744 Ki > 10000 nM T58589 COK10P 57402745 Ki > 10000 nM T58589 CGW59E 57403174 IC50 = 78 nM T58589 CW5O2D 57403175 IC50 = 188 nM T58589 CT6PB0 57403390 IC50 = 1.32 nM T58589 C9KLZ4 57403391 IC50 = 0.86 nM T58589 CG0VE7 57403503 Ki > 10000 nM T58589 CT74HP 57403504 Ki > 10000 nM T58589 CWO85L 68867798 Ki = 3.5 nM T58589 C69UHS 68868627 Ki = 5.8 nM T58589 C79JCF 68868975 Ki = 10 nM T58589 CP8FI7 68869351 Ki = 34 nM T58589 C06EMT 68869570 Ki = 3.3 nM T58589 C0VL1X 68869647 Ki = 0.8 nM T58589 CP0O3A 68870388 Ki = 4.7 nM T58589 CJ5XU4 70683374 Ki = 138 nM T58589 C3X0JV 70685470 Ki = 481 nM T58589 C2O3AY 70685471 Ki = 1 nM T58589 CP7QY1 70687620 Ki = 3.8 nM T58589 C6Z9WM 70688994 Ki = 2300 nM T58589 CXHO48 70688995 Ki = 59 nM T58589 CXAC04 70689675 Ki = 480 nM T58589 C49OIX 70691811 Ki = 1400 nM T58589 C13AMV 70691812 Ki = 6.3 nM T58589 C61JIR 70691813 Ki = 628 nM T58589 CKHP92 70691814 Ki = 2.9 nM T58589 CMV3F0 70692051 IC50 > 10000 nM T58589 C03TXD 70693872 Ki = 166 nM T58589 CZ41AD 70693873 Ki = 4.3 nM T58589 C0YZ2D 70695304 Ki = 2300 nM T58589 CL41AT 70695989 Ki = 2.2 nM T58589 CUX47G 71449505 IC50 = 2500 nM T58589 C6B0OV 71450888 Ki > 10000 nM T58589 C8YG2E 71454501 Ki = 1.8 nM T58589 CTIA35 71454502 Ki = 2.6 nM T58589 CHMG56 71456247 Ki = 7.1 nM T58589 CK01OM 71459890 Ki > 10000 nM T58589 C3Z7AR 71719128 Ki < 0.2 nM T58589 CJ2I4X 73346673 IC50 > 10000 nM T58589 C4QLS2 73346675 IC50 > 10000 nM T58589 CE1WK4 73348186 IC50 = 3019.95 nM T58589 CS27DN 73348187 IC50 = 1621.81 nM T58589 C2GO9F 73349741 IC50 > 10000 nM T58589 CNBL34 73351264 IC50 > 10000 nM T58589 CT72YC 73351265 IC50 > 10000 nM T58589 CO7W1C 73354242 IC50 = 389.05 nM T58589 CF49RH 73354498 Ki = 0.9 nM T58589 CDX4V9 73354499 Ki = 24 nM T58589 CUK4W3 73355813 IC50 = 4570.88 nM T58589 CWMR48 76331576 Ki = 0.023 nM T58589 C61FVX 90662943 Ki = 0.035 nM T58589 CSW30M 90662945 Ki > 10 nM T58589 CYEV01 137640759 IC50 = 4040 nM T58589 CRX0E4 137657568 IC50 = 2000 nM T58589 D00FAE 44316621 Ki = 5.6 nM T58589 D00FUT 123884 Ki = 382 nM T58589 D02DGP 44316161 Ki = 0.22 nM T58589 D04KFR 9831083 Ki = 8 nM T58589 D04WHO 9916412 Ki = 0.0078 nM T58589 D05TZN 122227 Ki < 0.2 nM T58589 D0L3GT 16108961 Ki = 0.7 nM T58589 D0N2GM 44316620 Ki = 83 nM T58589 D0U4SG 10281725 Ki = 85 nM T58589 D0V0LY 5310951 IC50 = 990 nM T62815 D01XYJ 35370 Ki = 150000 nM T62815 D0D1AL 3559 Ki = 590000 nM T62815 D0Y3KG 3121 Ki = 1600000 nM T62815 CF8W5U 68929 Ki = 162000 nM T62815 C57YCN 640695 IC50 = 507000 nM T62815 C2XI6Z 6971242 IC50 = 513000 nM T62815 CM4KP8 6971243 IC50 = 275000 nM T62815 CLI53U 6976566 IC50 = 214000 nM T62815 CX3B2N 6976567 IC50 = 130000 nM T62815 C16OIX 6976568 IC50 = 105000 nM T62815 C1CLV4 6976569 IC50 = 79000 nM T62815 CM6UB5 6992933 IC50 = 532000 nM T62815 C7RVQ1 7004960 IC50 = 344000 nM T62815 CBYR84 7058027 IC50 = 518000 nM T62815 CCAZ92 7058028 IC50 = 337000 nM T62815 C2D6MG 7058029 IC50 = 489000 nM T62815 C2JAE6 11491985 IC50 = 225000 nM T62815 CQJ29R 11513913 IC50 = 651000 nM T62815 C9VD3N 11550148 IC50 = 599000 nM T62815 C9PD1C 11557377 IC50 = 366000 nM T62815 C5XLW0 11564555 IC50 = 284000 nM T62815 C8LDV4 11607933 IC50 = 394000 nM T62815 CEFO25 11615192 IC50 = 179000 nM T62815 CCO5B8 11629630 IC50 = 317000 nM T62815 CD08XY 11636907 IC50 = 166000 nM T62815 CL1A3Y 11643947 IC50 = 540000 nM T62815 CP4ZE5 11658372 IC50 = 158000 nM T62815 CI5WQ9 11708159 IC50 = 301000 nM T62815 CX67NF 11715277 IC50 = 351000 nM T62815 CV3TC0 11831435 IC50 = 2000 nM T62815 C5VS2K 12328973 Ki = 113000 nM T62815 CQ47CA 12328974 IC50 = 182000 nM T62815 CNA17L 12337217 Ki = 301000 nM T62815 CA0M7Q 15148407 Ki = 101000 nM T62815 CR2I5A 16719568 IC50 = 4000 nM T62815 CCIK89 16720943 IC50 = 10000 nM T62815 C3XL7S 16720946 IC50 = 5000 nM T62815 CVS98C 17749637 IC50 = 5000 nM T62815 CE3O7S 18503890 IC50 = 500 nM T62815 C9RJD7 18503891 IC50 = 600 nM T62815 C50QKO 18503892 IC50 = 200 nM T62815 C1CT0N 18503893 IC50 = 400 nM T62815 CGO9E8 18503894 IC50 = 200 nM T62815 CC61VS 18503895 IC50 = 900 nM T62815 CN9FM4 18503899 IC50 = 500 nM T62815 CNS15Y 18503900 IC50 = 3000 nM T62815 CCS8Y9 18503901 IC50 = 16000 nM T62815 C29BLC 18503902 IC50 = 32000 nM T62815 CF72UR 18503905 IC50 = 800 nM T62815 CO63PD 18503907 IC50 = 3000 nM T62815 C30EWI 18503908 IC50 = 900 nM T62815 C3ZYJ1 18503909 IC50 = 400 nM T62815 C9EZF1 18503911 IC50 = 10000 nM T62815 C59OUH 18503912 IC50 = 18000 nM T62815 CHS8L5 18503913 IC50 = 4000 nM T62815 CSW96O 18503915 IC50 = 300 nM T62815 CHU60D 18503916 IC50 = 500 nM T62815 CXBU90 18503917 IC50 = 300 nM T62815 CB36RZ 18503918 IC50 = 400 nM T62815 CR9F0S 18503919 IC50 = 400 nM T62815 CDE1G2 18503920 IC50 = 800 nM T62815 C53NHK 18503921 Ki = 18.4 nM T62815 C5XMF7 18523698 IC50 = 900 nM T62815 CJ8XY0 18523699 IC50 = 700 nM T62815 CM6R0L 18523707 IC50 = 2000 nM T62815 CARN24 18523708 IC50 = 3000 nM T62815 CX8IJ4 18523709 IC50 = 12000 nM T62815 C7D5BX 18523710 IC50 = 8000 nM T62815 CCX5K6 18523711 IC50 = 41000 nM T62815 C2XMT1 18523712 IC50 = 1000 nM T62815 CGX30S 18523713 IC50 = 300 nM T62815 C69YMN 18523714 IC50 = 13000 nM T62815 CS28DQ 18523716 IC50 = 28000 nM T62815 CA9R0S 18523717 IC50 = 3000 nM T62815 C9LE0F 18523719 IC50 = 200 nM T62815 CBOW96 18523720 IC50 = 200 nM T62815 C87YIX 18523721 IC50 = 200 nM T62815 C25YFP 44423322 IC50 = 500 nM T62815 CULW28 44423323 IC50 = 700 nM T62815 CA34IP 89826402 IC50 > 300000 nM T62815 CZE16B 146026197 IC50 > 50000 nM T62815 D0M7YB 12311096 IC50 = 100 nM T62815 D0Z8EV 446541 Ki = 1500 nM T98264 D03DXN 66435 IC50 > 300000 nM T98264 D0I2AN 86298439 IC50 = 1440 nM T98264 CW68ZS 61672 IC50 = 2630 nM T98264 C7KJ3B 114917 IC50 = 1970 nM T98264 C5X1YU 160254 IC50 = 39500 nM T98264 C4IRY2 164676 IC50 = 2140 nM T98264 CCEG90 259329 IC50 = 40400 nM T98264 CONR62 444765 Ki = 350000 nM T98264 C9B3YM 444766 Ki > 2000000 nM T98264 CM0IQ3 446665 IC50 = 31000 nM T98264 C5Y3DJ 446871 Ki = 289000 nM T98264 C7GU8T 470607 IC50 = 12360 nM T98264 CELG48 998012 IC50 = 38760 nM T98264 CJ90PO 1159989 IC50 = 85000 nM T98264 CB7OS1 2964738 IC50 = 160000 nM T98264 C3NL9W 3246406 IC50 = 68000 nM T98264 C35LZP 4774445 Ki = 100000 nM T98264 CPM09B 5327156 IC50 = 203000 nM T98264 C4BE0F 9874843 IC50 = 9000 nM T98264 COX2J8 9930943 IC50 = 19000 nM T98264 CA75NG 9985013 IC50 = 15000 nM T98264 C3A8JL 10256983 IC50 = 6300 nM T98264 CZTN01 10675368 IC50 = 5000 nM T98264 CT4H0O 11006141 IC50 = 16000 nM T98264 C1JAC5 11425923 IC50 = 3670 nM T98264 C5K9MX 17748269 Ki = 17000 nM T98264 C3TV7F 19779154 IC50 = 129000 nM T98264 C54IUM 21778115 IC50 > 50000 nM T98264 C1OR3D 22084082 Ki = 28000 nM T98264 CDTE90 24180456 IC50 = 4000 nM T98264 C21ECL 24180507 Ki = 9700 nM T98264 CE9B6H 25014222 IC50 > 20000 nM T98264 C1Y0KM 25101546 Ki = 14000 nM T98264 CZ4M3C 25141412 IC50 = 15000 nM T98264 C4WM9S 25262527 IC50 = 15700 nM T98264 C3P8XN 42644186 IC50 > 40000 nM T98264 C98IOF 42644187 IC50 > 40000 nM T98264 CL04IU 44156271 IC50 = 14000 nM T98264 C1V7WS 44334321 Ki = 29000 nM T98264 CEL2Q6 44334377 Ki > 200000 nM T98264 CT20HY 44359237 Ki = 60000 nM T98264 C5YV1R 44359299 Ki > 2000000 nM T98264 C76DPK 44387848 EC50 = 50000 nM T98264 C36CRP 44387849 EC50 = 150000 nM T98264 CXU27L 44401026 EC50 = 50000 nM T98264 CZ6S7W 44401113 EC50 = 85000 nM T98264 CXL68A 44401147 EC50 = 160000 nM T98264 CGHV34 44401148 EC50 = 70000 nM T98264 CZC37T 44401149 EC50 = 140000 nM T98264 C01BYZ 44401229 EC50 = 80000 nM T98264 CL9BV8 44401230 EC50 = 180000 nM T98264 C7ABG4 44401231 EC50 = 220000 nM T98264 CLU5N2 44434676 IC50 = 38000 nM T98264 CWN8V5 44434677 IC50 = 13000 nM T98264 CA9X5W 44434678 IC50 = 9000 nM T98264 CY4LH6 44434679 IC50 = 25000 nM T98264 CBUP13 44434680 IC50 = 12000 nM T98264 C3R2HL 44563278 IC50 = 12640 nM T98264 CR50UK 44563344 IC50 = 27380 nM T98264 C9PC6L 44563345 IC50 = 5200 nM T98264 C3HDB9 44563372 IC50 = 4080 nM T98264 CT94FG 44563387 IC50 = 710 nM T98264 CDP45M 44563447 IC50 = 4050 nM T98264 C8MXT3 44563448 IC50 = 890 nM T98264 C7MP5Y 44563570 IC50 = 6000 nM T98264 C5Q2FM 44563588 IC50 = 126000 nM T98264 C7D5GS 44563589 IC50 = 140000 nM T98264 CBV8J9 44563590 IC50 = 78000 nM T98264 CP2H1Y 44563591 IC50 = 231000 nM T98264 CHNU48 44563656 IC50 = 10000 nM T98264 C3LMP9 44563657 IC50 = 6000 nM T98264 CO1GI5 45482833 Ki = 2200 nM T98264 CYRC54 45482878 IC50 > 40000 nM T98264 CK98JB 45482885 IC50 > 40000 nM T98264 CQ5U3C 45482886 IC50 > 40000 nM T98264 C8Z7HX 45482894 IC50 > 40000 nM T98264 CCKE09 45482895 IC50 > 40000 nM T98264 C1ULD8 45483667 Ki = 94000 nM T98264 CLGB06 46830252 IC50 > 10000000 nM T98264 C81CPM 46861833 IC50 = 10600 nM T98264 C0A9LD 46861834 IC50 = 9790 nM T98264 C2IU1Z 49796692 IC50 = 61000 nM T98264 CSBV96 50898774 IC50 = 3000 nM T98264 C4AEZ1 50925509 IC50 = 378 nM T98264 C95QWO 50925510 IC50 = 335 nM T98264 CK1YX2 50941649 IC50 = 5760 nM T98264 C1PJL0 50941745 IC50 = 408 nM T98264 CRF1O3 50942131 IC50 = 486 nM T98264 C2NJ3B 51003508 IC50 = 14000 nM T98264 CMDB84 53316640 IC50 > 50000 nM T98264 C9GVU5 53317937 IC50 > 50000 nM T98264 CV4QD5 53317938 IC50 = 17700 nM T98264 CWT10N 53319270 IC50 > 50000 nM T98264 CRC82E 53320578 IC50 > 50000 nM T98264 C8Y4KW 53320579 IC50 = 25700 nM T98264 CF35GK 53320580 IC50 = 18500 nM T98264 C04CYS 53320581 IC50 > 50000 nM T98264 CBI29Z 53321875 IC50 = 53100 nM T98264 C94WKB 53324565 IC50 > 50000 nM T98264 CCNG89 54576098 IC50 = 9840 nM T98264 CV3YH5 54576318 IC50 = 26500 nM T98264 C4CAU1 54576319 IC50 = 2430 nM T98264 CYK80P 54576320 IC50 = 16340 nM T98264 CKD3W9 54576321 IC50 = 10970 nM T98264 C1P4QM 54576322 IC50 = 13020 nM T98264 C1GDN4 54768308 IC50 = 15550 nM T98264 C1VCJ9 54768351 IC50 = 18500 nM T98264 CF7X2K 54768352 IC50 = 13220 nM T98264 C48KOI 54768353 IC50 = 12500 nM T98264 CK3W0Z 54768391 IC50 = 10720 nM T98264 C01LRT 54768392 IC50 = 16440 nM T98264 CNZY43 56589511 IC50 > 10000000 nM T98264 C53XYO 56589513 IC50 > 10000000 nM T98264 CHM5V3 56660070 IC50 > 120000 nM T98264 CHOF39 56670422 IC50 > 120000 nM T98264 CI9R8M 56670423 IC50 > 120000 nM T98264 CL3N0K 56673907 IC50 > 120000 nM T98264 CAL96I 56673908 IC50 > 120000 nM T98264 CEK3S2 56680547 IC50 > 120000 nM T98264 C72JTU 56681854 IC50 = 68900 nM T98264 CJ50EL 56681855 IC50 = 52600 nM T98264 CN3EW7 56683882 IC50 > 120000 nM T98264 C5CQY2 56683883 IC50 > 120000 nM T98264 CV4PW2 56683884 IC50 = 40400 nM T98264 CZP28F 57327772 IC50 = 24450 nM T98264 CG71TE 57380427 IC50 > 10000000 nM T98264 C4QJD7 57380429 IC50 > 10000000 nM T98264 CLTX25 57380431 IC50 > 10000000 nM T98264 CU94DW 57380433 IC50 = 129000 nM T98264 CCY75L 57380662 IC50 > 10000000 nM T98264 CE24LJ 57380664 IC50 = 167000 nM T98264 CWZ9E2 57380666 IC50 > 10000000 nM T98264 C9H7GI 57380668 IC50 > 10000000 nM T98264 CXW05S 57390693 IC50 > 10000000 nM T98264 CE57HQ 57395972 IC50 > 10000000 nM T98264 CGC16T 57397768 IC50 > 10000000 nM T98264 C18FTX 57397769 IC50 > 10000000 nM T98264 CQNG21 57397770 IC50 > 10000000 nM T98264 CX3A5R 57399431 IC50 > 10000000 nM T98264 CU5ND3 57514697 IC50 = 21000 nM T98264 C2BT9H 70673568 IC50 = 5000 nM T98264 C3AJ7H 70981706 IC50 = 2300 nM T98264 CP4H6L 70981726 IC50 = 2300 nM T98264 C2KS7Y 70982811 IC50 = 2490 nM T98264 C7VES4 71449486 IC50 = 16810 nM T98264 C5XB2N 71456091 IC50 > 100000 nM T98264 CP43AS 71461531 IC50 > 100000 nM T98264 CXI0F3 71561559 IC50 > 100000 nM T98264 CE0Y3O 71561685 IC50 = 4900 nM T98264 C3M4CF 71561686 IC50 = 4200 nM T98264 C82KCZ 71561687 IC50 = 3400 nM T98264 CDA8P2 71561688 IC50 = 34000 nM T98264 C87EXF 71561689 IC50 = 2600 nM T98264 CP9HX5 71561815 IC50 = 760 nM T98264 C9H5YS 71561816 IC50 = 5700 nM T98264 C61MWP 71561817 IC50 = 5100 nM T98264 C9GO5M 71561818 IC50 = 11500 nM T98264 CWA30F 71561819 IC50 = 5300 nM T98264 CBC4G0 71561820 IC50 = 7100 nM T98264 CPV8Y3 71561944 IC50 = 3700 nM T98264 CPWU40 71597177 IC50 > 50000 nM T98264 CT4MK9 71717989 IC50 > 100000 nM T98264 CCY15D 71734765 IC50 = 910 nM T98264 CS0XU2 72163288 IC50 = 10910 nM T98264 C6F1TD 72163289 IC50 = 14050 nM T98264 C0FWS2 72163422 IC50 = 24370 nM T98264 C2RNH4 72163424 IC50 = 17940 nM T98264 CNLB62 72163425 IC50 = 15770 nM T98264 C2JNO9 73345604 EC50 = 75000 nM T98264 C68EIC 73351713 EC50 = 60000 nM T98264 C20TML 73351714 EC50 = 140000 nM T98264 C1DWU4 73353952 IC50 = 7530 nM T98264 C9UP3V 73353954 IC50 = 12640 nM T98264 CS5O4J 73355491 IC50 = 6930 nM T98264 CMDC47 73357035 IC50 = 8790 nM T98264 CY0K7L 73357036 IC50 = 10610 nM T98264 CT1JH8 86766297 IC50 = 18180 nM T98264 CL4IN3 86766306 IC50 = 17760 nM T98264 CBK96X 90666455 IC50 > 20000 nM T98264 C61PBQ 90666456 IC50 > 20000 nM T98264 C40WCO 90666457 IC50 > 20000 nM T98264 C2ZGE9 90666458 IC50 > 20000 nM T98264 CG5TY1 90666459 IC50 > 20000 nM T98264 CWQN87 90666460 IC50 > 20000 nM T98264 CLU52N 90666461 IC50 = 15020 nM T98264 C0DW7A 90666462 IC50 > 20000 nM T98264 CXMC74 90666463 IC50 > 20000 nM T98264 C19JKD 101884098 IC50 = 78000 nM T98264 CX81PZ 118706101 IC50 = 6.8 ug.mL-1 T98264 CV5Q8J 118706102 IC50 = 5.1 ug.mL-1 T98264 CX2A8G 118722143 IC50 > 120000 nM T98264 CV5F0I 118722144 IC50 > 120000 nM T98264 C32ODE 118729111 IC50 = 5130 nM T98264 CTV62N 118729112 IC50 = 38420 nM T98264 CP9E4Q 118729113 IC50 = 19250 nM T98264 CS2XI7 118729114 IC50 = 8670 nM T98264 C3LN4T 118729115 IC50 = 10000 nM T98264 CF9KD7 118729116 IC50 = 9210 nM T98264 C27YKT 118729117 IC50 = 9250 nM T98264 C5FXC0 118729118 IC50 = 23650 nM T98264 C90UMX 118729119 IC50 = 24880 nM T98264 C4XZ2J 118729123 IC50 = 32240 nM T98264 C5GM1D 118729125 IC50 = 11120 nM T98264 CHF7U0 118729126 IC50 = 15680 nM T98264 C0IJ2X 118737463 IC50 = 8000 nM T98264 CN02HB 122182193 IC50 = 2310 nM T98264 CI87OL 122182194 IC50 = 9080 nM T98264 C12OHP 122187565 IC50 = 7300 nM T98264 CXHR32 122187566 IC50 = 4800 nM T98264 C59OUG 122187567 IC50 = 6000 nM T98264 CKT67D 122196241 IC50 = 2310 nM T98264 C2PVC5 122196288 IC50 = 9610 nM T98264 CV2H8T 122196290 IC50 = 11360 nM T98264 C46PST 127024952 IC50 > 120000 nM T98264 CF05SB 127025572 IC50 > 120000 nM T98264 C0KDZ2 127025573 IC50 > 120000 nM T98264 CI0NR9 127025574 IC50 > 120000 nM T98264 C6RI3J 127025575 IC50 > 120000 nM T98264 C5Z4PH 127025576 IC50 > 120000 nM T98264 C94EIF 127025577 IC50 > 120000 nM T98264 CR87HW 127025578 IC50 > 120000 nM T98264 CM9CP5 127027398 IC50 > 120000 nM T98264 C2A4GS 127027399 IC50 > 120000 nM T98264 CYOQ30 127027703 IC50 > 120000 nM T98264 CX52UN 127027704 IC50 > 120000 nM T98264 C6TIJ1 127027705 IC50 > 120000 nM T98264 C6H9SE 127027706 IC50 > 120000 nM T98264 C2X4JK 127027707 IC50 > 120000 nM T98264 C6UR4C 127027724 IC50 > 120000 nM T98264 C0RQ1U 127027725 IC50 > 120000 nM T98264 C0K2UI 127028022 IC50 > 120000 nM T98264 C1WA5T 127028346 IC50 > 120000 nM T98264 CC8HW0 127028347 IC50 > 120000 nM T98264 C6T0DY 127028683 IC50 > 120000 nM T98264 CL6QV7 127028684 IC50 > 120000 nM T98264 CG68NT 127028685 IC50 > 120000 nM T98264 C3MCH5 127028686 IC50 > 120000 nM T98264 CIAX67 127050086 IC50 = 2450 nM T98264 CEL9C4 127052247 IC50 = 6460 nM T98264 CF5HN6 132938289 IC50 = 8800 nM T98264 CZC42X 135924009 IC50 = 27700 nM T98264 C5BL1Z 135924010 IC50 = 103700 nM T98264 C9UA3N 135924011 IC50 = 32600 nM T98264 C1V8JE 135924012 IC50 = 7100 nM T98264 C8HP1O 135924013 IC50 = 18000 nM T98264 CHUD85 135924014 IC50 = 18100 nM T98264 CTZ5K1 135924015 IC50 = 15900 nM T98264 CAF8B6 135924016 IC50 = 32400 nM T98264 CK4X8S 135924017 IC50 = 10800 nM T98264 CE1FB0 135924018 IC50 = 122800 nM T98264 C39EPD 135924019 IC50 = 43100 nM T98264 CEH2M5 135924020 IC50 = 74200 nM T98264 CN6I5O 135924021 IC50 = 72500 nM T98264 CKW8X5 135924023 IC50 = 19400 nM T98264 CO3EX1 135924024 IC50 = 15700 nM T98264 CBJ7F8 135924025 IC50 = 40900 nM T98264 C81SHP 135924026 IC50 = 42500 nM T98264 CI62JU 135924027 IC50 = 60800 nM T98264 CAL83P 135924028 IC50 = 18300 nM T98264 CJ14VX 135924029 IC50 = 73400 nM T98264 C5C4EP 135924030 IC50 = 15400 nM T98264 C5QIK7 137174949 IC50 > 120000 nM T98264 CDZN68 137635090 IC50 = 10600 nM T98264 C28DUQ 137642390 IC50 = 34620 nM T98264 C48YBW 137646377 IC50 = 5290 nM T98264 CRU6Z7 137796282 IC50 = 72720 nM T98264 C0WMZ4 139593950 IC50 > 36800 nM T98264 C6NQ9I 145720956 IC50 = 14000 nM T98264 C4DWG8 145950748 IC50 = 3450 nM T98264 CIZE64 145960181 IC50 = 2940 nM T98264 CT6I5O 145961409 IC50 = 1090 nM T98264 C58OBV 145971193 IC50 = 850 nM T98264 CUE85W 145971302 IC50 = 4280 nM T98264 CV3FS9 145972458 IC50 = 8630 nM T98264 CB2I5V 155517051 IC50 = 2800 nM T98264 CGUP05 155517773 IC50 = 1520 nM T98264 C1HL4K 155519234 IC50 = 2800 nM T98264 CZ75SL 155521073 IC50 = 2950 nM T98264 C2WP6O 155522824 IC50 = 2800 nM T98264 CW1V5X 155522892 IC50 = 2800 nM T98264 CQ63GA 155537698 IC50 = 1110 nM T98264 CRU6F2 155538623 IC50 = 3990 nM T98264 C3Y6ZF 155538861 IC50 = 29900 nM T98264 CRH8J5 155548680 IC50 = 2540 nM T98264 CL1S9J 155565716 IC50 = 5160 nM T98264 C7W5HT 155566457 IC50 = 27100 nM T98264 D01BZE 73659 IC50 > 40000 nM T98264 D07LUJ 64945 IC50 = 25780 nM T98264 D0E0BU 444763 Ki = 16000 nM T98264 D0F9RO 6918774 IC50 = 24560 nM T98264 D0SJ2Q 10494 IC50 = 14190 nM T98264 D0U8IF 10114 IC50 = 65400 nM T98264 D0Y1RO 1829 Ki = 80000 nM T98264 D0Y5SB 444764 Ki = 510000 nM T48195 D06YPU 39912 IC50 = 100 nM T48195 D00QKI 9865554 IC50 = 16 nM T48195 D0LJ1B 9838712 IC50 = 5.3 nM T48195 D0ZL4F 180540 IC50 = 34 nM T48195 CNB6V7 114864 IC50 = 110 nM T48195 CMJ91Y 667550 IC50 = 50 nM T48195 CCVO02 9972278 IC50 = 360 nM T48195 C1L2WF 10018018 IC50 > 20000 nM T48195 CG2F7V 10200589 IC50 = 398 nM T48195 C7M8NX 10267982 IC50 = 42 nM T48195 C2BM1R 10402760 IC50 = 110 nM T48195 CC7T5M 11414892 IC50 = 80 nM T48195 C6H5VS 11625425 IC50 = 40 nM T48195 CYU1N8 12146502 IC50 = 46 nM T48195 CP6C4M 15980787 IC50 = 43 nM T48195 CT2D7W 15980830 IC50 = 410 nM T48195 CWEK41 15980918 IC50 > 20000 nM T48195 CM31SA 15980919 IC50 = 5100 nM T48195 C2OW0T 15981315 IC50 = 760 nM T48195 CV5M7D 15981316 IC50 = 160 nM T48195 CEW06X 15981317 IC50 = 200 nM T48195 C9KT1A 15981347 IC50 = 220 nM T48195 CY79RO 15981348 IC50 = 94 nM T48195 CT4C8A 15981349 IC50 = 50 nM T48195 CFJ3N8 15981350 IC50 = 680 nM T48195 CQGO53 16098481 IC50 = 251 nM T48195 C5NPO3 44284796 IC50 = 83 nM T48195 CCZ79T 44285113 IC50 > 20000 nM T48195 CO2Z4F 44285114 IC50 > 20000 nM T48195 C7CAM3 44285230 IC50 = 1000 nM T48195 C9VTS1 44285279 IC50 = 220 nM T48195 C30HNE 44285280 IC50 = 2700 nM T48195 CA52QI 44285430 IC50 = 12500 nM T48195 CFA7G2 44298268 Ki = 23000 nM T48195 CK45QG 44298269 Ki = 1700 nM T48195 CX7RL3 44298270 Ki = 68000 nM T48195 CVB2L1 44298317 Ki = 300 nM T48195 C6AE8K 44298340 Ki = 10000 nM T48195 CM3NT2 44298341 Ki = 13000 nM T48195 CKEX94 44298371 Ki = 120000 nM T48195 C6Q3WF 44298372 Ki = 190000 nM T48195 CAY2Q5 44298412 Ki = 750000 nM T48195 C3V1OQ 44298415 Ki = 3100000 nM T48195 C4EZ1W 44298416 Ki = 1850000 nM T48195 CAZG75 44298417 Ki = 890000 nM T48195 CWJX62 44298478 Ki > 1000 nM T48195 CEPB90 44298479 Ki > 1000 nM T48195 CWIA49 44298480 Ki > 30000 nM T48195 C8A9ZY 44298517 Ki > 30000 nM T48195 CRB25O 44298566 Ki = 55000 nM T48195 C5HB7Q 44298567 Ki = 27000 nM T48195 CE1FD5 44298568 Ki = 400000 nM T48195 C8WR7Q 44298569 Ki = 61000 nM T48195 C46FCX 44298606 Ki = 265000 nM T48195 CY3NW7 44298652 Ki = 155000 nM T48195 CK15HY 44298653 Ki = 15000 nM T48195 C06XVP 44298672 Ki = 62000 nM T48195 CED36R 44298676 Ki = 42000 nM T48195 C7QI1B 44298677 Ki = 29000 nM T48195 C6IW4P 44298701 Ki = 14000 nM T48195 C0QCP8 44298702 Ki = 5000 nM T48195 CL8E5P 44298703 Ki = 107000 nM T48195 C37RPZ 44298719 Ki = 42000 nM T48195 CO40US 44298729 Ki = 32000 nM T48195 C91FYI 44298730 Ki = 49000 nM T48195 CYI87G 44298744 Ki = 55000 nM T48195 C0RV8X 44298745 Ki = 27000 nM T48195 CUGS48 44298788 Ki = 28000 nM T48195 CY58NT 44298789 Ki = 2050000 nM T48195 CIZ42J 44298801 Ki = 2700000 nM T48195 C7RS5H 46896782 IC50 = 52 nM T48195 CX57UB 46896783 IC50 = 80 nM T48195 C0CEV2 46897163 IC50 = 22 nM T48195 C8E3GN 46897164 IC50 = 1220 nM T48195 CPL1N2 46897165 IC50 = 90 nM T48195 CI2J0B 46897254 IC50 = 387 nM T48195 CV7HR1 46897255 IC50 = 689 nM T48195 CE2D6V 77844109 IC50 > 10000 nM T48195 CC7Y9A 77844110 IC50 > 10000 nM T48195 C0VD5A 122187268 IC50 = 185 nM T48195 CW51VO 135485575 IC50 = 8990 nM T48195 C6J7ZP 135673987 IC50 = 2000 nM T48195 D09FHA 11322291 IC50 = 1.8 nM T48195 D09MAZ 46897162 IC50 = 36 nM T40332 D04AIT 5280445 Ki = 10100 nM T40332 D0FT4R 107706 Ki = 37 nM T40332 D0K8KX 5280343 Ki = 11900 nM T40332 D0SH3I 387447 Ki = 2300 nM T40332 D0V3YT 10324367 IC50 = 17000 nM T40332 D0X7JN 5280980 IC50 < 40000 nM T40332 D0X9CH 3010818 IC50 = 680 nM T40332 D00LOB 9866964 Ki > 26000 nM T40332 D06KJQ 42601552 IC50 > 30000 nM T40332 D08PBB 177992 IC50 = 23 nM T40332 D0A0SI 66601502 IC50 = 0.065 nM T40332 D0U2BH 65064 IC50 = 12800 nM T40332 D0VO0T 24800541 IC50 = 3550 nM T40332 D0Y6SQ 2536 IC50 > 100000 nM T40332 D00AWA 9938355 Ki = 0.013 nM T40332 D02PHE 46861623 IC50 = 12 nM T40332 D02YSI 44316902 Ki = 12 nM T40332 D06DET 9807572 IC50 = 29 nM T40332 D08ZCW 9910174 IC50 > 10 nM T40332 D0I0FM 44445940 Ki = 10 nM T40332 D0R9ON 65837 IC50 = 1000 nM T40332 D0U7OU 3220 IC50 = 52000 nM T40332 D0WY9H 9892148 Ki = 1.3 nM T40332 C19TYR 44343121 IC50 = 10500000 nM T40332 C3N6FP 44342779 IC50 = 13500000 nM T40332 CT8RD6 1526 Ki = 15 nM T40332 CX09SM 1636 Ki = 18 nM T40332 C7ET4R 6773 IC50 = 39000 nM T40332 C4RT3E 10208 IC50 = 18000 nM T40332 C73JPZ 10639 IC50 = 6200 nM T40332 C0WN5U 13926 Ki = 9549.93 nM T40332 CE1GQ3 68236 Ki = 4786.3 nM T40332 CF7O4D 125700 IC50 = 40 nM T40332 CB17TY 128954 IC50 = 2000 nM T40332 CLX4V7 130395 IC50 > 100000 nM T40332 C5Q7EX 160817 IC50 = 11000 nM T40332 CW4AE7 178662 Ki = 0.014 nM T40332 C0Z8UG 191187 IC50 = 10000 nM T40332 CIGP91 196813 IC50 = 9000 nM T40332 CQJD84 216294 Ki = 12 nM T40332 C05PDV 223000 Ki = 831763.77 nM T40332 C4HLA8 223062 IC50 = 100000 nM T40332 CC9E0Y 232547 IC50 = 15600 nM T40332 CPJW07 294660 Ki = 4365.16 nM T40332 CH46ID 296003 Ki = 1778.28 nM T40332 C1WRQ6 309231 IC50 >= 28000 nM T40332 CXOC26 339156 Ki = 112.2 nM T40332 CB39JK 343129 IC50 = 13000 nM T40332 CJ1R7C 433517 IC50 > 100000 nM T40332 CCX8A5 468714 Ki = 6 nM T40332 CT79FC 468715 IC50 = 44 nM T40332 CG2SL7 468760 IC50 = 92 nM T40332 C5XV2G 481422 IC50 > 1000000 nM T40332 CW1KP3 481437 IC50 > 300000 nM T40332 C7ZUS1 481440 IC50 > 600000 nM T40332 C9EAL6 482277 IC50 > 75000 nM T40332 C58PLQ 482278 IC50 > 75000 nM T40332 C2G9IH 482279 IC50 > 75000 nM T40332 C5L4ED 482280 IC50 > 75000 nM T40332 CTW1J9 482282 IC50 > 75000 nM T40332 CK0O9U 482283 IC50 > 75000 nM T40332 CX0SQ5 482284 IC50 > 75000 nM T40332 C6Y5SA 482285 IC50 > 75000 nM T40332 C2D7MH 482286 IC50 > 75000 nM T40332 CAZV26 482287 IC50 > 75000 nM T40332 C2QP9I 482288 IC50 > 75000 nM T40332 C3L9TI 482289 IC50 > 75000 nM T40332 CO3N0A 482290 IC50 > 75000 nM T40332 CZ15KR 482291 IC50 > 75000 nM T40332 C0HV7G 482292 IC50 > 75000 nM T40332 CC1RP8 483672 IC50 < 60 nM T40332 C3N7CD 487110 IC50 = 30000 nM T40332 C6B1KZ 504659 Ki = 6.457 nM T40332 CVE0Y8 504661 Ki = 0.1148 nM T40332 CTD7X8 504663 Ki = 0.04266 nM T40332 CN67CR 555078 Ki = 28 nM T40332 C32HXT 589588 Ki = 1905.46 nM T40332 CRQ98S 589620 Ki = 645.65 nM T40332 CM7T6V 589629 Ki = 302 nM T40332 C9Y3FN 589883 Ki = 10964.78 nM T40332 C9YWX0 607716 IC50 = 16000 nM T40332 C0LDK9 611090 Ki = 7244.36 nM T40332 CD23NS 628877 IC50 >= 28000 nM T40332 CFO5M9 630168 IC50 >= 28000 nM T40332 CQ94TR 639465 Ki = 15700 nM T40332 CD5P8N 644145 IC50 = 5000 nM T40332 CTDG97 644152 IC50 = 168000 nM T40332 CAJ4F5 644153 IC50 = 21000 nM T40332 C7Q0UO 644154 IC50 = 41000 nM T40332 CREX84 644155 IC50 = 151000 nM T40332 C28PBX 644930 IC50 > 100000 nM T40332 CCKZ79 668744 IC50 = 51500 nM T40332 C53FNM 674593 Ki = 15 nM T40332 C45NBS 674629 Ki = 107 nM T40332 C21HDC 674632 Ki = 24 nM T40332 CG2UK8 674633 Ki = 1000 nM T40332 CX1W4S 674635 Ki = 7200 nM T40332 C9PI4L 674639 Ki = 9000 nM T40332 C3M8OE 674640 Ki = 9000 nM T40332 CI9LH0 674642 Ki = 1100 nM T40332 CBX3U0 674652 Ki = 6 nM T40332 COD8V2 674657 Ki = 3100 nM T40332 CW5ZA1 680939 Ki = 24 nM T40332 CN06WE 685663 Ki = 10700 nM T40332 CXDC18 714833 Ki = 24500 nM T40332 CFP1A9 730175 Ki = 820 nM T40332 C87WLA 753830 Ki = 50900 nM T40332 C0ER8S 767161 IC50 = 124900 nM T40332 CDVJ42 767163 IC50 = 15500 nM T40332 CE10WO 776842 IC50 = 160200 nM T40332 CYF3T7 806239 Ki = 8912.51 nM T40332 CU85MI 823661 Ki = 2884.03 nM T40332 C8BQU5 833517 Ki = 300 nM T40332 C2O5LR 849299 IC50 = 20000 nM T40332 CLR3H1 899247 Ki = 21 nM T40332 CV23JB 914899 Ki = 169.82 nM T40332 C5SN4P 928297 Ki = 3630.78 nM T40332 CLR10O 928795 Ki = 11.48 nM T40332 CQ2R0M 1011274 IC50 = 78300 nM T40332 C5AM9V 1169804 IC50 > 100000 nM T40332 CWJL58 1169805 IC50 > 100000 nM T40332 CX1W4I 1170184 IC50 > 100000 nM T40332 C2PRY6 1269450 IC50 = 6700 nM T40332 CUL5Y4 1331170 IC50 > 100000 nM T40332 CW90DG 1457429 IC50 > 100000 nM T40332 CENL04 1523065 IC50 = 5100 nM T40332 CYH46M 1993219 IC50 > 100000 nM T40332 C0D8LM 2213207 Ki = 29900 nM T40332 CO4AB7 2264784 IC50 = 52200 nM T40332 C3A9BT 2302435 Ki = 1.8 nM T40332 C8DW1C 2372853 IC50 > 100000 nM T40332 CC5R9U 2796528 Ki = 34673.69 nM T40332 CKJ5T0 2812522 IC50 = 61 nM T40332 CYW3M6 3223864 IC50 > 100000 nM T40332 C45ZIU 3368775 IC50 >= 28000 nM T40332 CAEW98 3435549 IC50 > 100000 nM T40332 CNJM56 3534338 IC50 > 60000 nM T40332 CPC72H 3835811 IC50 = 32100 nM T40332 CJDR03 3963048 Ki = 1600 nM T40332 C6JF0O 4155991 IC50 = 2700 nM T40332 C9FTM3 5113707 Ki = 71 nM T40332 C9UOQ3 5151183 Ki = 2570.4 nM T40332 CF9VK2 5236960 IC50 = 26900 nM T40332 CK2X1T 5271294 IC50 > 75000 nM T40332 CWIC65 5279637 IC50 = 36100 nM T40332 CAF61Z 5289347 Ki = 25 nM T40332 CV20QH 5294946 IC50 > 100000 nM T40332 CO58XD 5311161 IC50 > 100000 nM T40332 CA63CX 5367020 Ki = 8128.31 nM T40332 CCUM24 5467627 IC50 = 2900 nM T40332 C4VIT3 5480997 IC50 = 20 nM T40332 CDV72G 5480998 IC50 = 3200 nM T40332 CZ1XU5 5876194 IC50 = 19600 nM T40332 COD34R 6451966 Ki = 954.99 nM T40332 CQS5E1 6888904 IC50 = 17600 nM T40332 C8OE6S 6913584 IC50 > 100000 nM T40332 CG2A7X 7028541 IC50 = 84800 nM T40332 CECO04 8967103 IC50 >= 28000 nM T40332 CF4TK5 8967105 IC50 >= 28000 nM T40332 C89JBK 9636571 IC50 > 100000 nM T40332 CZ8V7U 9799757 IC50 = 1000 nM T40332 CE56CV 9804093 Ki = 114 nM T40332 CUX59Q 9804457 Ki = 0.066 nM T40332 CL8TN0 9806936 Ki = 170 nM T40332 CRJ6I2 9808548 Ki = 1.66 nM T40332 C4DIG6 9808564 Ki = 0.022 nM T40332 C84XOY 9808874 Ki = 0.025 nM T40332 C92HSW 9809309 IC50 = 24 nM T40332 CZ6W1Y 9809577 IC50 = 21 nM T40332 CFSX09 9815828 Ki = 1.5 nM T40332 CT2WM1 9827187 Ki = 4.9 nM T40332 C4I0UG 9829396 IC50 = 6.6 nM T40332 C9YO0Z 9830006 Ki = 0.7 nM T40332 CH31WN 9830037 Ki = 0.008 nM T40332 CGNB60 9830581 IC50 = 9500 nM T40332 CR54JK 9830622 IC50 = 30 nM T40332 CZFT64 9830860 IC50 = 20 nM T40332 C6NIU3 9831417 Ki = 0.2 nM T40332 CM53FA 9834041 Ki = 63000 nM T40332 C2NX3Q 9852363 IC50 = 27 nM T40332 C6R7XS 9852378 IC50 = 23 nM T40332 CDL5O0 9866692 Ki = 0.7 nM T40332 CBC5V7 9866842 Ki = 0.035 nM T40332 CX92DE 9871592 Ki = 26 nM T40332 CI5T7N 9873436 IC50 = 17 nM T40332 C2T6QH 9875205 Ki = 0.45 nM T40332 CS3C0L 9887581 IC50 < 150 nM T40332 CL61HY 9888442 Ki = 0.014 nM T40332 CG2EZ0 9889108 Ki = 0.31 nM T40332 C3H0LQ 9892781 Ki = 3.35 nM T40332 CCX4N0 9893147 Ki = 170 nM T40332 COA8T5 9894208 IC50 = 6.6 nM T40332 CEO04L 9894378 Ki = 5.1 nM T40332 CZQ97P 9895636 IC50 = 14 nM T40332 C9IZB4 9904055 IC50 = 4000 nM T40332 C7KJP3 9908917 Ki = 1.73 nM T40332 C1T5VN 9912574 Ki = 725 nM T40332 CJ6M8N 9915812 IC50 > 300000 nM T40332 C08KHW 9917190 IC50 = 62 nM T40332 C2HY9N 9917412 IC50 = 47 nM T40332 CQ84MG 9917430 Ki = 6.3 nM T40332 C8D5CH 9920598 Ki = 51 nM T40332 CGT3K4 9932145 Ki = 0.16 nM T40332 CRK8F2 9933704 Ki = 44.3 nM T40332 CG2Q1F 9934160 Ki = 79.7 nM T40332 CA8DY4 9938068 IC50 = 28 nM T40332 CXA7B4 9953653 Ki = 0.3 nM T40332 C3EPC4 9955758 Ki > 22000 nM T40332 CUY4S5 9960766 IC50 = 27 nM T40332 C2VU3Y 9962219 IC50 = 84 nM T40332 C2CE1A 9962331 Ki = 0.2 nM T40332 C3HI6E 9972080 IC50 = 47 nM T40332 CM06CQ 9973338 Ki = 100 nM T40332 C1UKM3 9977679 Ki = 320 nM T40332 C4J0GP 9978440 Ki = 52 nM T40332 CW56ZP 9978595 Ki = 500 nM T40332 C1VB6K 9980302 Ki = 0.6 nM T40332 C7E9BA 9980407 Ki = 54 nM T40332 C5ZNO7 9980554 Ki = 43 nM T40332 C58VXC 9982602 Ki = 51 nM T40332 C09EYT 9983109 Ki = 94 nM T40332 C12ITA 9984374 Ki = 190 nM T40332 C2B9IN 9985199 Ki = 13 nM T40332 CME79C 9985374 Ki = 25 nM T40332 CIJ5L2 9987080 IC50 = 6700 nM T40332 CCE26Y 10002661 Ki = 0.03 nM T40332 CPO47T 10002668 Ki = 46 nM T40332 C7UON4 10002900 Ki = 270 nM T40332 C6ANW0 10004044 Ki = 280 nM T40332 C7YSW2 10004682 Ki = 340 nM T40332 CW2G0I 10005629 Ki = 261 nM T40332 CMV31E 10006663 Ki = 4300 nM T40332 CBXZ29 10007724 Ki = 13 nM T40332 CC1JY8 10008607 Ki = 4.2 nM T40332 CTEQ15 10008826 Ki = 0.55 nM T40332 C95FMS 10009631 Ki = 1.5 nM T40332 CFBX35 10014336 IC50 > 1000000 nM T40332 C1MKH6 10015569 IC50 > 1000000 nM T40332 CI8PL9 10016936 IC50 = 221.5 nM T40332 CN16OT 10022457 Ki = 8 nM T40332 C87NHX 10023592 Ki = 1100 nM T40332 CWB04G 10023940 IC50 = 28000 nM T40332 CO75QM 10024023 Ki = 0.8 nM T40332 CHC6E8 10024782 Ki = 101 nM T40332 CH32TU 10026529 Ki = 6.5 nM T40332 CPMA30 10026572 IC50 = 200 nM T40332 CEO32W 10027816 Ki = 9.3 nM T40332 CG0H4T 10028039 Ki = 10 nM T40332 CL1RN4 10028081 Ki = 19 nM T40332 C6GMX9 10028968 Ki > 500000 nM T40332 CQ9A2O 10029003 Ki = 7.7 nM T40332 C9XH3K 10029428 Ki = 49 nM T40332 CL8WU9 10029465 Ki = 1.2 nM T40332 CEA89V 10029470 Ki = 270 nM T40332 CDM5V2 10029484 Ki = 0.8 nM T40332 CEN3S7 10029919 Ki = 15 nM T40332 CF1SN8 10029970 Ki = 33 nM T40332 C07UYT 10030271 Ki = 66 nM T40332 C1KIE7 10030460 Ki = 21000 nM T40332 CYW21E 10030835 Ki = 20 nM T40332 CGK82S 10031500 Ki = 88 nM T40332 CUM1S3 10032109 Ki = 12 nM T40332 C1FM9L 10032899 Ki = 0.33 nM T40332 C35XZA 10036576 Ki = 257.04 nM T40332 C8RNZ5 10043396 Ki = 60 nM T40332 CG7F8T 10048188 Ki = 210 nM T40332 CVHQ60 10048700 Ki = 22 nM T40332 CEH7X8 10049090 Ki = 6.2 nM T40332 CS9U8H 10052095 Ki = 80000 nM T40332 C5HYK8 10052622 Ki = 130 nM T40332 CH3NT1 10052689 Ki = 300 nM T40332 CNK54H 10052690 Ki = 16 nM T40332 C14TNZ 10053504 Ki = 89 nM T40332 CH7B0C 10053891 Ki = 2.3 nM T40332 C4K3QL 10054085 Ki = 0.11 nM T40332 CVZU17 10054360 Ki = 0.07 nM T40332 CRJ2W9 10054620 Ki = 0.011 nM T40332 C8DHG9 10054626 Ki = 1.1 nM T40332 CH8YI6 10054689 Ki = 16 nM T40332 CF2V0Y 10055681 Ki = 0.3 nM T40332 CH70LT 10055869 Ki = 0.81 nM T40332 CRL8D2 10060710 Ki = 1.349 nM T40332 CM7XN1 10067940 Ki = 24 nM T40332 CO6QV4 10069016 Ki = 350 nM T40332 CBAU50 10071439 Ki = 4.9 nM T40332 CWJ29L 10071504 Ki = 3400 nM T40332 CIO8S2 10071747 Ki = 57 nM T40332 C8GVA0 10072025 Ki = 0.06 nM T40332 C7MZL9 10073426 Ki = 16 nM T40332 CVGW19 10074999 Ki = 22000 nM T40332 C4DG6S 10075424 Ki = 40 nM T40332 C8YT1B 10076039 Ki = 24 nM T40332 C8BHG0 10076168 Ki = 5600 nM T40332 C3WCV4 10076315 Ki = 87000 nM T40332 C5V1YC 10076625 Ki = 8.4 nM T40332 C8TVW3 10076806 Ki = 5.7 nM T40332 CL59QU 10076807 Ki = 42 nM T40332 C2H5PM 10076832 Ki = 330 nM T40332 C9MZ0X 10076908 Ki = 1.9 nM T40332 C6FUN8 10077271 Ki = 42 nM T40332 CZG6L4 10077327 Ki = 4.4 nM T40332 C67HUG 10077412 Ki = 0.2 nM T40332 CO4NR6 10077495 Ki = 2.8 nM T40332 CMG13S 10077534 Ki = 0.4 nM T40332 C1CFV6 10078395 Ki = 0.43 nM T40332 C7CW1P 10080504 IC50 = 58 nM T40332 CD3N9Q 10084731 Ki = 5.754 nM T40332 C45MKR 10087296 IC50 > 50000 nM T40332 CEH86P 10088912 Ki = 4 nM T40332 CKX3J8 10092679 Ki = 0.07 nM T40332 C5YF2B 10092898 Ki = 18 nM T40332 CEN06H 10093642 IC50 > 100000 nM T40332 CNS73M 10093670 IC50 = 140 nM T40332 CPSY01 10093766 Ki = 8.7 nM T40332 CZU18G 10094548 Ki = 730 nM T40332 CA6WS0 10095870 Ki = 1 nM T40332 CPY1Q7 10097512 Ki = 0.55 nM T40332 CNX98I 10098504 Ki = 6.6 nM T40332 CU4N0V 10098932 Ki = 3.6 nM T40332 CC7WV4 10099005 Ki = 8.2 nM T40332 CNZ68F 10099030 Ki = 22 nM T40332 CKM91H 10099223 Ki = 3.5 nM T40332 CWG0Q4 10099305 Ki = 8.5 nM T40332 CSXU07 10099653 Ki = 1.18 nM T40332 CP2D8N 10099715 Ki = 2.4 nM T40332 C83RTX 10100215 Ki = 0.37 nM T40332 C57PNI 10101455 Ki = 3 nM T40332 CSY56V 10101683 Ki = 0.66 nM T40332 CV8U6L 10101834 Ki = 0.1 nM T40332 C58BWQ 10113382 Ki = 14 nM T40332 C3VA2F 10116108 Ki = 6.38 nM T40332 C3RFT8 10118557 Ki = 2.55 nM T40332 CJLB36 10138967 Ki = 43.8 nM T40332 CXR76P 10138974 Ki = 16.6 nM T40332 CVBL74 10160118 Ki = 26.4 nM T40332 CG6Z3R 10165977 Ki = 1.37 nM T40332 CPU95M 10198315 Ki = 83.18 nM T40332 C5BEP1 10227093 Ki = 6.76 nM T40332 CD8OU0 10241309 Ki = 6900 nM T40332 CDLR68 10250073 Ki = 62 nM T40332 CUY45Q 10251702 Ki = 350 nM T40332 CEHC01 10254338 Ki = 8.5 nM T40332 CA3E1W 10256440 Ki = 8 nM T40332 CK1NB4 10257209 Ki = 34 nM T40332 CZ1B8M 10257257 Ki = 87 nM T40332 CY8NL9 10257279 Ki = 11 nM T40332 CKX95D 10257311 Ki = 6.6 nM T40332 CR8D4G 10257948 Ki = 0.93 nM T40332 CEC58D 10258115 Ki = 4.4 nM T40332 C04XJL 10264928 Ki = 13 nM T40332 CXWQ38 10274774 Ki = 23.5 nM T40332 CB28OA 10275675 Ki = 8.75 nM T40332 CA2YG9 10297988 Ki = 10.7 nM T40332 C97QRW 10298752 Ki = 15.3 nM T40332 CT3A2S 10300047 Ki = 24.8 nM T40332 C8DU7V 10300829 Ki = 2.25 nM T40332 C0X2CU 10302080 Ki = 0.52 nM T40332 CQA3X0 10321894 Ki = 0.023 nM T40332 CD5QM2 10323328 Ki = 39 nM T40332 CW8A4E 10325129 Ki = 52 nM T40332 CW3X4Q 10325189 Ki = 3400 nM T40332 CNXE05 10325233 Ki = 1.4 nM T40332 CA9X6O 10326668 Ki = 8000 nM T40332 CWV2A9 10327283 Ki = 25 nM T40332 C0PJN3 10331933 Ki = 2.73 nM T40332 COA7X1 10338134 Ki = 8 nM T40332 CYCO34 10341700 Ki = 0.07079 nM T40332 CU7FE3 10342642 Ki = 26 nM T40332 C0FME8 10343129 Ki = 27 nM T40332 CS16AL 10343238 Ki = 43000 nM T40332 CIE4G0 10343847 Ki = 3.59 nM T40332 C2GLK6 10346121 IC50 > 50000 nM T40332 C1PI8K 10346591 Ki = 150 nM T40332 C9GL1U 10346870 Ki = 15 nM T40332 CKJC76 10347501 Ki = 23 nM T40332 CO3WL8 10347655 Ki = 33 nM T40332 CC3NH2 10347721 Ki = 4.1 nM T40332 CZ58RW 10347871 Ki = 3.5 nM T40332 C0VL6K 10347891 Ki = 1.8 nM T40332 C1XV8P 10348077 Ki = 4.8 nM T40332 C2VWM9 10348957 Ki = 0.013 nM T40332 CMW89Q 10349323 Ki = 36 nM T40332 C6YUW8 10349541 Ki = 25 nM T40332 CY3L2F 10358434 Ki = 31 nM T40332 C1B6UP 10361206 Ki = 2800 nM T40332 C2I1XM 10363347 Ki = 51000 nM T40332 CK60UV 10366641 Ki = 15 nM T40332 C7K9PJ 10367217 Ki = 2500 nM T40332 CE6VW2 10368099 Ki = 6.7 nM T40332 CS4UX5 10368963 Ki = 16000 nM T40332 C62KEB 10369593 Ki = 4 nM T40332 CK2YU1 10369681 Ki = 4.5 nM T40332 C01CPM 10369682 Ki = 480 nM T40332 CATB56 10370141 Ki = 31 nM T40332 CU3ZF4 10370563 Ki = 8.1 nM T40332 CAT02C 10370853 Ki = 1.8 nM T40332 CGH83D 10371178 Ki = 3.8 nM T40332 CH1RY5 10371190 Ki = 150000 nM T40332 CG9UT0 10371325 Ki = 1.3 nM T40332 CC7RW2 10371949 Ki = 43 nM T40332 CDP4T7 10372563 Ki = 0.5 nM T40332 C5FYM0 10372900 Ki = 0.2 nM T40332 CND9F2 10378134 Ki = 12.59 nM T40332 C1P9VJ 10389512 Ki = 42 nM T40332 CKY94N 10389844 Ki = 34 nM T40332 C8I3WV 10390162 IC50 = 20300 nM T40332 C6RHB5 10390443 Ki = 48 nM T40332 CL49JD 10391720 Ki = 13 nM T40332 CMZ05N 10391723 Ki = 15 nM T40332 CX0KM7 10392329 IC50 = 1 nM T40332 CD6MQ8 10392657 Ki = 5.6 nM T40332 C2FLG8 10392960 Ki = 79 nM T40332 CF05VG 10393052 Ki = 71 nM T40332 C48IQH 10393970 Ki = 47 nM T40332 CH32ZO 10394405 Ki = 32 nM T40332 C3TU6O 10394985 Ki = 25 nM T40332 CBF97Q 10397988 Ki = 91 nM T40332 CC5Q6K 10405508 Ki = 15000 nM T40332 CL48XK 10412920 Ki = 80 nM T40332 C4IUT8 10414698 Ki = 0.011 nM T40332 CSDZ76 10414749 Ki = 30 nM T40332 CPE67V 10414810 Ki = 11 nM T40332 CSH83N 10414990 Ki = 40 nM T40332 C36VYB 10415426 Ki = 12000 nM T40332 CHV37A 10415461 Ki = 15 nM T40332 CQY79A 10415479 Ki = 6.9 nM T40332 CSKX23 10415744 Ki = 17 nM T40332 CNT27F 10415810 Ki = 60 nM T40332 CN7D3W 10415869 Ki = 12 nM T40332 C4MC7H 10416037 Ki = 9.4 nM T40332 C2KJR0 10426076 Ki = 2700 nM T40332 C3IC8F 10432526 Ki = 1100 nM T40332 CW2D3O 10432804 Ki = 1000 nM T40332 CTF92S 10434048 Ki = 37 nM T40332 C84QZG 10434385 Ki = 28 nM T40332 C0CPI1 10435585 Ki = 23 nM T40332 C1RI4C 10435834 Ki = 6.6 nM T40332 CK2SL0 10435916 Ki = 170 nM T40332 C1Z6TU 10436952 Ki = 48 nM T40332 COST60 10436956 Ki = 7 nM T40332 CV7YC6 10436990 Ki = 320 nM T40332 CH6Q2J 10437166 Ki = 6 nM T40332 CV1LD0 10437728 Ki = 18 nM T40332 CXR12A 10438569 Ki = 42 nM T40332 C59OXM 10439034 Ki = 20 nM T40332 C5N0OZ 10439282 Ki = 0.35 nM T40332 C5Z1IB 10440161 Ki = 0.66 nM T40332 C79OYK 10440316 Ki = 0.1 nM T40332 C08TPL 10440405 Ki = 0.06 nM T40332 CQ5DM6 10452703 Ki = 1.995 nM T40332 CQ6G5E 10453174 Ki = 290 nM T40332 CHNG31 10453578 Ki = 1.995 nM T40332 COX97B 10454399 Ki = 30 nM T40332 CJ5FS1 10456006 Ki = 26 nM T40332 CTF5G1 10457246 Ki = 6100 nM T40332 CW7FT8 10457506 Ki = 40 nM T40332 CRH7I5 10457598 Ki = 71 nM T40332 C06QJW 10457653 IC50 > 50000 nM T40332 CKY0C5 10459649 Ki = 8.8 nM T40332 C6BQL9 10459820 Ki = 57 nM T40332 C5N9DB 10460031 IC50 > 300000 nM T40332 C1L0VN 10460376 Ki = 23 nM T40332 CB4K1S 10460522 Ki = 11 nM T40332 COL58Y 10460549 Ki = 18 nM T40332 CQ0S8Y 10460720 Ki = 9 nM T40332 CH17CO 10460911 Ki = 1.1 nM T40332 C15YVO 10461918 IC50 = 33 nM T40332 CO1XS4 10462803 Ki = 9.4 nM T40332 CHJ27G 10462942 Ki = 0.65 nM T40332 C9Y2MK 10468056 Ki = 1.43 nM T40332 CYD67S 10475537 Ki = 0.1 nM T40332 C8C9YS 10477377 Ki = 26 nM T40332 C7DHG4 10478230 Ki = 510 nM T40332 CCNA48 10479704 Ki = 360 nM T40332 CO6U0V 10479967 Ki = 20.5 nM T40332 C9XB8D 10481065 Ki = 17 nM T40332 CJNT56 10481404 Ki = 190 nM T40332 C09HJD 10481557 Ki = 410 nM T40332 C5U6DL 10481845 Ki = 469 nM T40332 C2GEQ9 10482544 Ki = 52 nM T40332 CR5F0K 10483274 Ki = 9.6 nM T40332 CU0EA3 10483607 IC50 = 260000 nM T40332 C90THX 10484261 Ki = 4.6 nM T40332 CWN6L8 10484563 Ki = 72 nM T40332 CF5W6B 10491098 Ki = 133 nM T40332 CFP53Y 10502109 IC50 = 2260 nM T40332 C60MXW 10505465 Ki = 0.027 nM T40332 CQW51O 10506703 IC50 = 183000 nM T40332 CYQB28 10507021 IC50 > 300000 nM T40332 CFNK35 10507077 IC50 > 300000 nM T40332 CPET76 10517251 Ki = 238 nM T40332 CA4RW1 10517868 IC50 = 11000 nM T40332 CG34WR 10518548 Ki = 100 nM T40332 C5Y1XO 10527174 Ki = 0.5 nM T40332 CYJ58Q 10528103 Ki = 15 nM T40332 CQES53 10529707 Ki = 130 nM T40332 C84WLX 10531366 Ki = 5.7 nM T40332 CQC62W 10531634 Ki = 1.6 nM T40332 CZ29RX 10537951 Ki = 3.981 nM T40332 C7B8LG 10549313 Ki = 0.85 nM T40332 C5J7MX 10550886 Ki = 4281 nM T40332 C5KO9W 10553305 Ki = 0.81 nM T40332 C5G6SC 10553739 Ki = 15 nM T40332 CAKY60 10554399 Ki = 3 nM T40332 C7NJQ1 10554839 IC50 > 300000 nM T40332 C0T6QD 10556018 Ki = 5500 nM T40332 CER1M4 10560388 Ki = 41.69 nM T40332 CC2DB8 10564561 Ki = 12.59 nM T40332 CVX74R 10569244 IC50 < 200 nM T40332 CP1HE3 10571766 Ki = 0.06 nM T40332 C6Y1XV 10573143 Ki = 0.03 nM T40332 C3F4KN 10577308 Ki = 12 nM T40332 C9EK8W 10579293 Ki = 1100000 nM T40332 CJ5MB0 10579493 Ki = 0.35 nM T40332 C3VR0Q 10579612 Ki = 1.1 nM T40332 C3HJ4N 10579613 Ki = 3.4 nM T40332 CXF17L 10579679 Ki = 3.1 nM T40332 CBM4L7 10591621 IC50 > 1000000 nM T40332 C7HM6O 10599457 Ki = 0.22 nM T40332 CZB90H 10601497 Ki = 330 nM T40332 CQ9BP2 10601989 Ki = 4200 nM T40332 CGS56E 10610038 Ki = 5.61 nM T40332 CKN60O 10612715 Ki = 51 nM T40332 CQ38DS 10615154 IC50 = 6600 nM T40332 CYQC10 10615902 IC50 = 1200 nM T40332 C53MHY 10616362 Ki = 288.4 nM T40332 CPN7X5 10624194 Ki = 11.8 nM T40332 C8XA3U 10626170 Ki = 8 nM T40332 CDLP35 10628028 Ki = 70 nM T40332 CS18WR 10635550 Ki = 5.7 nM T40332 COL8B0 10636536 Ki = 91 nM T40332 CG69CZ 10638623 IC50 = 36000 nM T40332 CD86WR 10647120 Ki = 0.72 nM T40332 CDL36E 10647461 Ki = 0.14 nM T40332 CQ0O5J 10648323 Ki = 160 nM T40332 C5T8WG 10650026 Ki = 57.8 nM T40332 CZ78MR 10651388 Ki = 9.9 nM T40332 CME37Y 10651433 Ki = 6.4 nM T40332 CBHW74 10653967 Ki = 1000 nM T40332 CMXS14 10653995 Ki = 20 nM T40332 CW75PO 10661946 IC50 > 500 nM T40332 CM2IJ0 10665528 IC50 = 75000 nM T40332 CQAG87 10670178 Ki = 0.025 nM T40332 C71RBG 10670907 Ki = 0.025 nM T40332 CX36QE 10671458 Ki = 0.034 nM T40332 CJ1B0W 10671534 Ki = 0.013 nM T40332 CDB35L 10673162 Ki = 74 nM T40332 CP1V5D 10673918 Ki = 44 nM T40332 CN0I1R 10673962 Ki = 2.3 nM T40332 CCF8L6 10674356 IC50 > 300000 nM T40332 COSG14 10675303 Ki = 58 nM T40332 C8A0EJ 10680902 Ki = 28.84 nM T40332 COM2A7 10687511 IC50 = 900 nM T40332 CVCW48 10694581 Ki = 310 nM T40332 CC35DA 10695507 IC50 = 2660 nM T40332 CNEA57 10696461 Ki = 42 nM T40332 CT6ME5 10696947 Ki = 19 nM T40332 CZ8C2D 10697242 Ki = 0.64 nM T40332 CGR40J 10697956 Ki = 12 nM T40332 CC2G9E 10698640 Ki = 14000 nM T40332 C8BX1N 10710010 IC50 = 25000 nM T40332 C2SK5B 10718228 Ki = 690 nM T40332 CH1B5D 10727846 Ki = 130 nM T40332 C2UGD0 10728016 Ki = 34.67 nM T40332 CY0B3X 10729570 Ki = 5.74 nM T40332 CB2ZE0 10732420 Ki = 204.17 nM T40332 CNK38E 10733818 Ki = 17.78 nM T40332 CMBL13 10738994 Ki = 910 nM T40332 C58TAI 10739339 Ki = 0.18 nM T40332 CWZ92Y 10741446 Ki = 0.11 nM T40332 CL7RC5 10742017 IC50 = 1440 nM T40332 CV6D9X 10744508 Ki = 0.9 nM T40332 C3MXP5 10744523 Ki = 16 nM T40332 CZC57E 10744893 Ki = 22 nM T40332 C5VGC3 10744962 Ki = 3.4 nM T40332 C3L7VF 10745054 Ki = 21 nM T40332 C7AEI6 10745144 IC50 > 300000 nM T40332 CZAT51 10747107 Ki = 18 nM T40332 CZP63T 10756289 IC50 > 75000 nM T40332 CB7V0K 10763054 Ki = 14 nM T40332 CL20BQ 10765017 Ki = 0.09 nM T40332 CLU87Q 10765018 Ki = 0.078 nM T40332 CR6S4Z 10767409 Ki = 13.9 nM T40332 CB50RU 10768396 Ki = 0.85 nM T40332 C0EC3Z 10769317 Ki = 8.9 nM T40332 CE38KS 10769657 Ki = 4.1 nM T40332 CZG97S 10783016 IC50 = 300 nM T40332 CEMV61 10786746 Ki = 0.05 nM T40332 CWM1X4 10788924 Ki = 0.21 nM T40332 CV0O8I 10789380 Ki = 0.25 nM T40332 CS9F4X 10789763 Ki = 5.8 nM T40332 C97TFC 10791626 Ki = 230 nM T40332 C0WZ5S 10792102 Ki = 15 nM T40332 CD4P6H 10793294 Ki = 8.4 nM T40332 C1NK2I 10793641 Ki = 0.35 nM T40332 CT56CL 10793708 Ki = 1.7 nM T40332 C7K4RS 10794780 Ki = 100 nM T40332 CIC52D 10799209 Ki = 10.7 nM T40332 C20LYK 10799960 Ki = 446.68 nM T40332 CH0TA1 10805857 IC50 = 3000 nM T40332 CFHQ20 10813515 Ki = 29.1 nM T40332 C0H9BP 10815491 Ki = 0.058 nM T40332 C3L1DQ 10815914 Ki = 0.38 nM T40332 CL0E8T 10816188 Ki = 7.5 nM T40332 C28DOK 10816650 IC50 > 300000 nM T40332 CGP01V 10817508 IC50 > 300000 nM T40332 CG9B1J 10819798 Ki = 1300 nM T40332 C04IOW 10827508 Ki = 43.65 nM T40332 CDN04R 10831749 Ki = 0.033 nM T40332 CJ9FT6 10832773 Ki = 0.052 nM T40332 CE9NM4 10835541 Ki = 0.083 nM T40332 CIHY04 10837647 Ki = 490 nM T40332 CGX75W 10839361 Ki = 100 nM T40332 CSK04U 10839694 Ki = 21.2 nM T40332 CP6S9N 10854087 IC50 = 200 nM T40332 C07UEM 10889772 Ki = 707.95 nM T40332 C9Q2XI 11230895 IC50 = 1900 nM T40332 C7CHR5 11236753 IC50 = 17000 nM T40332 CS0CP2 11247668 Ki = 11700 nM T40332 C92PMV 11253808 IC50 = 9900 nM T40332 CKPO36 11272981 IC50 = 0.9 nM T40332 C2M7UP 11343089 IC50 > 30000 nM T40332 C4VX3G 11534280 IC50 = 0.5 nM T40332 CLAK97 11540629 IC50 = 100000 nM T40332 CT4FV1 11563929 Ki = 5300 nM T40332 CD7JU2 11590336 IC50 = 6700 nM T40332 C7FV6O 11592854 Ki = 340 nM T40332 CV82NQ 11619625 IC50 = 44 nM T40332 C93USP 11626693 IC50 > 10000 nM T40332 CWQ25N 11741764 Ki = 2 nM T40332 CHS6B5 11742000 Ki = 2600 nM T40332 C6FBJ4 11742006 Ki = 17 nM T40332 CTFS51 11742114 Ki = 4.5 nM T40332 C6B2TV 11743404 Ki = 100 nM T40332 CB95LW 11754431 Ki = 6.1 nM T40332 CS1TC0 11754640 Ki = 0.08 nM T40332 CD5W1A 11755516 Ki = 70 nM T40332 C5EQ9D 11756768 Ki = 9.1 nM T40332 CD7E0H 11757806 Ki = 32 nM T40332 C34FJZ 11757887 Ki = 52 nM T40332 CSM9F4 11758548 Ki = 0.34 nM T40332 C53SEA 11760115 IC50 = 14000 nM T40332 CJ6IG2 11765406 Ki = 0.6 nM T40332 CFG62D 11777027 Ki = 56.23 nM T40332 CJ0E8V 11779851 IC50 = 610 nM T40332 CO6A8F 11795366 Ki = 620 nM T40332 CN7LE6 11796530 Ki = 36 nM T40332 C3BN8Q 11797855 Ki = 33 nM T40332 CW5KF3 11798332 Ki = 830 nM T40332 C7QM3S 11799612 Ki = 290 nM T40332 CYRC95 11800689 IC50 > 300000 nM T40332 CWK1G8 11801735 Ki = 0.35 nM T40332 C7L9FS 11802328 Ki = 150 nM T40332 CCNX57 11983863 IC50 = 36000 nM T40332 C4IYM7 12134435 IC50 = 62 nM T40332 C3TIQ7 12248312 Ki = 52 nM T40332 C4O9HJ 12290092 Ki = 7413.1 nM T40332 CU0RL3 12689300 IC50 = 4800 nM T40332 CN6Z8X 12689316 IC50 = 400 nM T40332 CI8BH7 12689319 IC50 = 50 nM T40332 CKQ0W6 12689323 IC50 = 20 nM T40332 C7DV9I 12689324 IC50 = 5700 nM T40332 CY0RD7 12689332 IC50 = 19000 nM T40332 C0OIN2 12735875 Ki = 64565.42 nM T40332 C0S1VX 12942058 IC50 = 1390000 nM T40332 C4O5EV 13129200 IC50 = 19000 nM T40332 C32VSL 13221326 Ki = 30902.95 nM T40332 C19FEY 13629121 IC50 = 2000 nM T40332 C41KQG 13629122 IC50 > 40000 nM T40332 CY0U2X 13629126 IC50 = 4000 nM T40332 C4LKW6 13787283 Ki = 933.25 nM T40332 CVJU63 13827088 Ki = 17.78 nM T40332 C73UJB 13827090 Ki = 4.898 nM T40332 C64HRM 13827091 Ki = 0.06761 nM T40332 C4UOW2 13827093 Ki = 0.1905 nM T40332 C8PBE1 13827094 Ki = 5.754 nM T40332 CG6L2Y 13849881 Ki = 75.5 nM T40332 CU6H5B 13849894 Ki = 144.54 nM T40332 C9HVJ5 13853503 Ki = 38.02 nM T40332 C7XH2D 13853505 Ki = 43 nM T40332 CUC1S9 13853506 Ki = 3600 nM T40332 CIN97K 13853507 Ki = 31622.78 nM T40332 C56YEI 13853508 Ki = 954.99 nM T40332 CYIJ53 13853509 Ki = 588.84 nM T40332 CBK13D 13853511 Ki = 22.91 nM T40332 CL28MT 13853512 Ki = 1995.26 nM T40332 CY8ZP3 13853515 Ki = 181.97 nM T40332 CSE35Q 13853516 Ki = 776.25 nM T40332 C8BC3R 13853517 Ki = 407.38 nM T40332 CM1F9R 13853519 Ki = 4.169 nM T40332 C1JYQ0 13853520 Ki = 0.9333 nM T40332 CKD31E 13853528 Ki = 5.888 nM T40332 CE17QS 13853530 Ki = 707.95 nM T40332 CSU9J2 13853531 Ki = 6.607 nM T40332 CHG37U 13853534 Ki = 147.91 nM T40332 CQK4T2 13853537 Ki = 20.89 nM T40332 CJO19A 13853538 Ki = 177.83 nM T40332 CG85UW 13853539 Ki = 239.88 nM T40332 C3YUS1 13853541 Ki = 37.15 nM T40332 C3KO7X 13853551 Ki = 18620.87 nM T40332 C50ERO 13853552 Ki = 66.07 nM T40332 CZ5R9T 13853553 Ki = 37.15 nM T40332 CV57RA 13853554 Ki = 169.82 nM T40332 CF2J8E 13853555 Ki = 46.77 nM T40332 CQ7SY6 13853556 Ki = 27.54 nM T40332 COV0G6 13853560 Ki = 12.02 nM T40332 C34BNK 13880838 IC50 = 40000 nM T40332 CXYN02 14010380 IC50 = 620 nM T40332 CKF19U 14010382 IC50 = 6200 nM T40332 C4P0AK 14010383 IC50 = 250 nM T40332 CZ16DP 14010384 IC50 = 1400 nM T40332 C6MY3O 14010385 IC50 = 19000 nM T40332 CAH1W7 14010386 IC50 = 6000 nM T40332 CUH75S 14010387 IC50 = 1000 nM T40332 C24WHI 14010388 IC50 = 850 nM T40332 C4Z5NT 14010389 IC50 = 800 nM T40332 CK5T2I 14010390 IC50 = 320 nM T40332 CGA68E 14010391 IC50 = 1500 nM T40332 C6CKZ7 14010392 IC50 = 350 nM T40332 C1C9FM 14010393 IC50 = 800 nM T40332 C15ACF 14010394 IC50 = 2200 nM T40332 C3QB5A 14010395 IC50 = 170 nM T40332 C7KV4T 14010396 IC50 = 12000 nM T40332 CFJ0O9 14010397 IC50 = 670 nM T40332 CF52UJ 14010398 IC50 = 150 nM T40332 C5ZVC9 14010399 IC50 = 900 nM T40332 CO6QD1 14010400 IC50 = 27 nM T40332 CZBO42 14010401 IC50 = 1500 nM T40332 C3S2KZ 14010402 IC50 = 55 nM T40332 C0Z8EN 14010403 IC50 = 84 nM T40332 C1VWO8 14010404 IC50 = 10000 nM T40332 CMS3V7 14010405 IC50 = 8000 nM T40332 CUT3S2 14010407 IC50 = 140 nM T40332 CPQ5N2 14010408 IC50 = 360 nM T40332 CT3HG6 14010410 IC50 = 460 nM T40332 CR27UM 14010411 IC50 = 1500 nM T40332 CY82DH 14010414 IC50 = 130 nM T40332 CFON34 14010415 IC50 = 450 nM T40332 CQ18TM 14010416 IC50 = 83 nM T40332 C59EVI 14010418 IC50 = 1800 nM T40332 CB8XQ1 14052374 IC50 = 10000 nM T40332 C87RMA 14089169 IC50 = 110 nM T40332 CS8BF9 14089170 IC50 = 100 nM T40332 CAF82P 14089172 IC50 = 300 nM T40332 CHZ75Q 14089173 IC50 = 210 nM T40332 C9KM6B 14089174 IC50 = 160 nM T40332 C5RWV4 14089175 IC50 = 1900 nM T40332 CUT74L 14089176 IC50 = 200 nM T40332 CO2C7I 14089177 IC50 = 5400 nM T40332 CAZM38 14089178 IC50 = 27 nM T40332 C2U7LD 14089179 IC50 = 100 nM T40332 C38RIF 14089180 IC50 = 8400 nM T40332 CGO1Q5 14089181 IC50 = 600 nM T40332 C68VEU 14089182 IC50 = 130 nM T40332 C5QE8G 14089184 IC50 = 80000 nM T40332 CQ3YT2 14089185 IC50 = 72 nM T40332 C7LBW3 14089186 IC50 = 9000 nM T40332 CXI47P 14089187 IC50 = 1000 nM T40332 C0A8HV 14207561 Ki = 0.4677 nM T40332 CUGW80 14207563 Ki = 0.3981 nM T40332 C0EIF7 14379792 IC50 > 40000 nM T40332 C3NK7L 14379796 IC50 = 60 nM T40332 CC9A3G 14379800 IC50 = 3000 nM T40332 CJFB97 14379803 IC50 = 30000 nM T40332 CCM8E6 14379806 IC50 = 2000 nM T40332 CGEU96 14488442 IC50 = 4000 nM T40332 CVI43O 14488443 IC50 > 40000 nM T40332 C3TG7L 14493342 Ki = 102 nM T40332 CC10KI 14513750 Ki = 3400 nM T40332 CV7A3W 14539951 Ki = 4300 nM T40332 C9G4DC 14542117 Ki = 512.86 nM T40332 C0AUT7 14760206 IC50 = 200 nM T40332 C1MR8P 14760208 IC50 = 500 nM T40332 CYC20A 14760210 IC50 = 100 nM T40332 CD1OC8 14760212 IC50 = 100 nM T40332 CG7J0I 14760231 IC50 = 800 nM T40332 CU3H5M 14760233 IC50 = 70 nM T40332 C2LS8V 14760235 IC50 = 100 nM T40332 C4SF7Z 14760237 IC50 = 200 nM T40332 CY76IR 14760239 IC50 = 100 nM T40332 CCNE24 14760241 IC50 = 400 nM T40332 C2A3HQ 14760243 IC50 = 40 nM T40332 C2FQ3E 14760247 IC50 = 400 nM T40332 C0P6KI 14760249 IC50 = 400 nM T40332 CY4HQ3 14760260 IC50 = 5000 nM T40332 C46LBG 14760262 IC50 = 100 nM T40332 CEZ3A4 14760264 IC50 = 800 nM T40332 CWK7S9 14760266 IC50 = 2000 nM T40332 CARP67 14760298 IC50 = 1000 nM T40332 CJ2HR7 14760300 IC50 = 200 nM T40332 CYJ3K2 14760306 IC50 > 50000 nM T40332 C5UP4K 14760308 IC50 > 50000 nM T40332 C5FVQ2 14760310 IC50 = 5000 nM T40332 CDW0S3 14760319 IC50 = 400 nM T40332 C0FA5S 14760334 IC50 = 430 nM T40332 CR6ZV5 14760337 IC50 = 2400 nM T40332 CL78BW 14760339 IC50 = 2230 nM T40332 CK3YT2 14760341 IC50 = 2330 nM T40332 C96RUH 14760343 IC50 = 1620 nM T40332 CBG83A 14760345 IC50 = 1820 nM T40332 CZO79G 14760347 IC50 = 630 nM T40332 C13ABK 14760351 IC50 = 940 nM T40332 C72HTW 14760353 IC50 = 910 nM T40332 CH7ZT3 14760355 Ki = 220 nM T40332 CZGD18 14760368 IC50 = 130 nM T40332 C4UM1D 14760370 IC50 = 1000 nM T40332 CBQ0Z1 14760376 IC50 = 1800 nM T40332 CAXH03 14760380 IC50 = 57800 nM T40332 C5F3MZ 14861885 IC50 = 3.7 ug.mL-1 T40332 COE37G 15035342 Ki = 290000 nM T40332 C3NM4I 15035343 Ki = 16500 nM T40332 CCWF97 15198479 IC50 = 6700 nM T40332 CQ0RU9 15200486 Ki = 28 nM T40332 C4Y8KR 15230194 Ki = 15 nM T40332 CG1NR2 15230196 Ki = 81 nM T40332 C1UH7S 15338151 Ki = 0.08 nM T40332 CT48FA 15407997 IC50 > 300000 nM T40332 CLGV32 15547238 IC50 > 10000 nM T40332 CN05KP 15573427 IC50 > 40000 nM T40332 CKR59B 15589985 IC50 > 10000000 nM T40332 CU1TD9 15726831 IC50 > 40000 nM T40332 C32CWO 15726832 IC50 > 40000 nM T40332 C6L5MJ 15726833 IC50 > 40000 nM T40332 CJQ6V7 15726835 IC50 > 40000 nM T40332 CAYS45 15726841 IC50 = 40000 nM T40332 C26CQI 15726842 IC50 > 40000 nM T40332 CVPL97 15726843 IC50 = 28000 nM T40332 CH7KS8 15726844 IC50 > 40000 nM T40332 CED5G0 15726845 IC50 = 1000 nM T40332 C0UYJ4 15726846 IC50 > 10000 nM T40332 C3VE9S 15726847 IC50 = 5000 nM T40332 CZG4F5 15726851 IC50 = 10000 nM T40332 CA4R1Z 15726852 IC50 = 36000 nM T40332 CSC4K3 15726857 IC50 = 300 nM T40332 C0YBI9 15726858 IC50 = 6000 nM T40332 CT6W4L 15726859 IC50 = 10000 nM T40332 C6TYB5 15726860 IC50 > 40000 nM T40332 CKJU90 15726861 IC50 = 10000 nM T40332 C8BD3T 15726862 IC50 = 6000 nM T40332 C3MIX7 15726863 IC50 = 1000 nM T40332 CRO39F 15726866 IC50 = 24000 nM T40332 C2EGD3 15726867 IC50 = 40000 nM T40332 CX1LM4 15726868 IC50 = 2000 nM T40332 CQY3B4 15726869 IC50 = 20000 nM T40332 CG9X0Z 15726871 IC50 > 40000 nM T40332 CO5MC2 15726874 IC50 > 40000 nM T40332 CYTK20 15726875 IC50 > 40000 nM T40332 CF49XE 15726876 IC50 = 4000 nM T40332 CDP91C 15743471 IC50 = 8700 nM T40332 CJ41CN 15743472 IC50 = 4200 nM T40332 C8YR1W 15743473 IC50 = 5900 nM T40332 CWU90T 15743474 Ki = 150 nM T40332 CZ6WU7 15838071 Ki = 5.47 nM T40332 COG9C4 15885812 Ki = 33.88 nM T40332 C5XRE1 15886812 Ki = 0.49 nM T40332 CPZU83 15928334 IC50 = 830 nM T40332 C72JFE 15955759 Ki = 251.19 nM T40332 C9M1EK 16104379 IC50 > 10000 nM T40332 CRQV57 16104920 IC50 = 49 nM T40332 C9OSM6 16144480 Ki = 120 nM T40332 CDR0G7 16145606 Ki = 100 nM T40332 CY20PW 16147332 Ki = 130 nM T40332 CF5Y3L 16147570 Ki = 8300 nM T40332 C7S6IT 16148231 Ki = 200 nM T40332 C0WX5C 16163030 Ki = 1300 nM T40332 CSXO69 16680454 IC50 = 352 nM T40332 C6AR3Q 16757019 IC50 = 316 nM T40332 CL8M0W 17755151 IC50 = 0.21 nM T40332 C0JBH9 18395047 IC50 > 50000 nM T40332 C2XTI9 18395048 IC50 > 50000 nM T40332 C63HAE 18572952 IC50 = 18000 nM T40332 CV86RX 18603196 Ki = 41 nM T40332 CRW81C 18607241 Ki = 1258.93 nM T40332 C50UPT 18607265 Ki = 870.96 nM T40332 C8MD2B 18607267 Ki = 213.8 nM T40332 CJ03UC 18633082 IC50 = 200 nM T40332 CZP68C 18633083 IC50 = 2000 nM T40332 CN85LE 18633087 IC50 = 200 nM T40332 CIYD09 18633089 IC50 = 10000 nM T40332 C3YRI4 18633090 IC50 = 150 nM T40332 CI9A1H 18643724 IC50 = 1330 nM T40332 CXF13I 18801003 IC50 > 5000 nM T40332 C7U4PY 19030591 Ki = 5.754 nM T40332 C7DPB4 19389555 Ki = 91.2 nM T40332 C6K1QN 19845653 Ki = 0.07079 nM T40332 CD4L1N 19845806 Ki = 0.2291 nM T40332 C5UDO2 20139259 Ki = 10 nM T40332 CRQ9Y6 20139310 Ki = 10 nM T40332 C1DRH4 20208290 Ki = 2818.38 nM T40332 CJ7TH3 20208319 Ki = 10.96 nM T40332 CP6UN4 20208423 Ki = 1348.96 nM T40332 C2M8AW 20208435 Ki = 16.98 nM T40332 CX59VG 20208455 Ki = 1202.26 nM T40332 CUG1K3 20208523 Ki = 645.65 nM T40332 CXHA26 21033975 Ki = 63 nM T40332 CGB92N 21731457 Ki = 109.65 nM T40332 C20KJO 21823504 Ki = 219 nM T40332 CD7CI2 22124919 Ki = 416.87 nM T40332 CS2X9Z 22152164 Ki = 77.62 nM T40332 CT58FO 22392859 IC50 > 10000000 nM T40332 CLU18Y 22881851 Ki = 28 nM T40332 CA2S6B 23151285 Ki = 1000 nM T40332 C5VSO2 23276168 Ki = 288403.15 nM T40332 CB63KH 23276169 Ki = 338844.16 nM T40332 C7QD8E 23276182 Ki = 346736.85 nM T40332 CR8LI0 23437569 Ki = 218.78 nM T40332 CUH0K4 23444468 Ki = 109.65 nM T40332 CS13PY 23657291 IC50 = 23 nM T40332 CTBO93 23664980 IC50 = 44 nM T40332 C9XJP3 23711928 IC50 = 3000 nM T40332 CBD3H5 23728722 Ki = 15 nM T40332 CN0VA7 24822701 IC50 > 50000 nM T40332 CW9D6P 24823445 Ki = 23.8 nM T40332 C2WI4S 24823446 Ki = 0.71 nM T40332 CU2O6S 24823609 Ki = 63.5 nM T40332 CT78NC 24854122 IC50 = 59100 nM T40332 CCD95H 24854123 IC50 = 71300 nM T40332 C9J2QD 24974797 Ki = 4570.88 nM T40332 C9TKJ6 24999408 IC50 = 390 nM T40332 CVI40X 24999724 IC50 = 93 nM T40332 C8G7FX 24999726 IC50 = 64 nM T40332 C8SNG4 25000364 IC50 = 110 nM T40332 C1UH4R 25000365 IC50 = 6000 nM T40332 C0GJ4N 25000368 IC50 = 8100 nM T40332 CUC8N5 25141405 IC50 = 3100 nM T40332 CX05JT 25205745 IC50 = 19 nM T40332 C3GS6F 33009902 IC50 > 10000 nM T40332 C2DEG7 42642360 IC50 < 0.3 nM T40332 CL0M7R 44143089 IC50 = 85113.8 nM T40332 CPT2B6 44266363 IC50 = 6100 nM T40332 CH9O7C 44266372 IC50 = 130 nM T40332 CX89JI 44266374 IC50 = 43000 nM T40332 C54FSU 44266698 IC50 = 110 nM T40332 CDS31V 44267097 Ki = 0.21 nM T40332 C9X4QL 44267147 Ki = 0.96 nM T40332 CUW9I2 44267176 Ki = 1.6 nM T40332 CR8O5J 44267221 Ki = 27 nM T40332 C97EWG 44267427 Ki = 1.2 nM T40332 C8EQ9C 44267442 Ki = 0.24 nM T40332 C43NJL 44267444 Ki = 0.17 nM T40332 C75REN 44267447 Ki = 0.47 nM T40332 C8QVJ6 44267462 Ki = 0.34 nM T40332 C3ZU7Q 44267468 Ki = 0.049 nM T40332 CMSI17 44272976 Ki = 19000 nM T40332 CN2X4F 44272977 Ki = 27000 nM T40332 CYV1W8 44273732 Ki = 270000 nM T40332 CFA21P 44273766 Ki = 190000 nM T40332 CNV18Y 44274239 Ki > 300000 nM T40332 CD84XF 44279475 IC50 > 50000 nM T40332 C0RQ3V 44279712 IC50 > 30000 nM T40332 CFJ2Z1 44279771 IC50 > 30000 nM T40332 C3IBQ0 44279792 IC50 > 50000 nM T40332 CQ57HR 44279823 IC50 > 50000 nM T40332 C5YF0J 44279873 IC50 > 50000 nM T40332 CROD68 44279951 IC50 > 50000 nM T40332 C6ZXK0 44280152 IC50 > 50000 nM T40332 CVZ54E 44280172 IC50 > 50000 nM T40332 C8D6VK 44282051 IC50 > 75000 nM T40332 CN7SA3 44287645 IC50 = 3900 nM T40332 C1GU7P 44287670 IC50 = 13000 nM T40332 C7QSK8 44287706 IC50 = 11000 nM T40332 CB8L9Q 44287782 IC50 = 8000 nM T40332 CR6QO0 44287881 IC50 = 6000 nM T40332 C5NR3Q 44287906 IC50 = 12000 nM T40332 CT98XO 44287910 IC50 = 5900 nM T40332 C3F9LM 44287918 IC50 = 21000 nM T40332 C42JSV 44287920 IC50 = 13000 nM T40332 C6AZV8 44287930 IC50 = 2500 nM T40332 C4KWZ8 44287967 IC50 = 6400 nM T40332 CR9YA8 44288052 Ki = 7500 nM T40332 C6KJ4D 44288060 IC50 = 6100 nM T40332 CMO3X2 44288136 IC50 = 4200 nM T40332 CDT93F 44288297 IC50 = 1300 nM T40332 CN04DK 44288315 Ki = 430 nM T40332 COP5H9 44288316 Ki = 1900 nM T40332 CJH40B 44295808 Ki = 17500 nM T40332 CSC8X9 44295983 Ki = 32 nM T40332 C6POB4 44296152 Ki = 0.7 nM T40332 CJC83Z 44296212 Ki = 13.6 nM T40332 C49ZTQ 44296213 Ki = 15 nM T40332 CNI4K8 44296327 Ki = 80 nM T40332 CSEG82 44296328 Ki = 2000 nM T40332 CA9R6Z 44296341 Ki = 60 nM T40332 CYO86L 44296343 Ki = 0.6 nM T40332 CWL62G 44296396 Ki = 3 nM T40332 CI0EM5 44296406 Ki = 32 nM T40332 C12XSO 44296649 Ki = 246 nM T40332 CN1I6M 44296666 Ki = 17.5 nM T40332 CJ37GI 44298562 Ki = 6.1 nM T40332 COB9F7 44298605 Ki = 0.41 nM T40332 C14GUD 44298619 Ki = 0.87 nM T40332 CKEA52 44298620 Ki = 1.8 nM T40332 CQAG41 44298819 Ki = 3.3 nM T40332 C6URN0 44298842 Ki = 43 nM T40332 CP50DO 44298855 Ki = 1.1 nM T40332 C94FOM 44298860 Ki = 1.7 nM T40332 CAK97H 44298884 Ki = 1.2 nM T40332 CMWF68 44298885 Ki = 5.4 nM T40332 CPN6G7 44298886 Ki = 60 nM T40332 CU8Z3V 44298888 Ki = 1.8 nM T40332 C0K2QM 44298908 Ki = 1.6 nM T40332 CGB10R 44298921 Ki = 4.2 nM T40332 CQ8B2N 44298922 Ki = 2 nM T40332 CT3DQ8 44298927 Ki = 55 nM T40332 C1FM8K 44298929 Ki = 2.7 nM T40332 C8U2WZ 44298945 Ki = 2.3 nM T40332 CO6MA7 44298966 Ki = 8 nM T40332 CUCW51 44298967 Ki = 10 nM T40332 CQGX12 44298970 Ki = 3.2 nM T40332 C62MQB 44298980 Ki = 2.5 nM T40332 C80XBS 44298984 Ki = 5.2 nM T40332 C4KTI6 44298990 Ki = 15 nM T40332 CB39FC 44298992 Ki = 11 nM T40332 C47SOH 44298993 Ki = 0.43 nM T40332 C2BYH3 44299001 Ki = 1.7 nM T40332 CGBR39 44299062 Ki = 190 nM T40332 CM54OT 44299064 Ki = 1.2 nM T40332 CIOE85 44299235 Ki = 12 nM T40332 CPO75N 44299253 Ki = 1.3 nM T40332 C8IL5V 44299896 IC50 = 36 nM T40332 C3A1YN 44299897 IC50 = 38 nM T40332 C5G6LV 44299976 IC50 = 15 nM T40332 CM24TU 44299977 IC50 = 24 nM T40332 C9G5QX 44299990 IC50 = 24 nM T40332 CZMJ96 44300040 IC50 = 18 nM T40332 CEW05I 44300059 IC50 = 59 nM T40332 CS28OU 44300070 IC50 = 0.1 nM T40332 CGE9W3 44300076 IC50 = 84 nM T40332 C69WJZ 44300092 IC50 = 30 nM T40332 C5FDJ3 44300093 IC50 = 36 nM T40332 C20JDX 44300119 IC50 = 40 nM T40332 CUKL54 44300133 IC50 = 43 nM T40332 C6V4XE 44300174 IC50 = 46 nM T40332 C6EU7G 44300177 IC50 = 38 nM T40332 C5G9KX 44300179 IC50 = 70 nM T40332 CV7F8N 44300180 IC50 = 34 nM T40332 C5RSX9 44300181 IC50 = 26 nM T40332 C30HJX 44300217 IC50 = 20 nM T40332 C9M3NU 44300289 IC50 = 46 nM T40332 COX87D 44304039 IC50 = 50 nM T40332 C68UDG 44306172 Ki = 320000 nM T40332 C6ZO2A 44306517 Ki = 1800000 nM T40332 CO42PE 44306533 Ki = 1000000 nM T40332 CY0M9E 44306778 IC50 = 40000 nM T40332 C51ZLR 44308482 Ki = 18 nM T40332 CZK3U8 44308945 Ki = 1.6 nM T40332 CKA3B8 44308946 Ki = 0.35 nM T40332 CF61VA 44308955 Ki = 0.81 nM T40332 C2Z9QB 44309043 Ki = 4.1 nM T40332 CQ80NX 44309049 Ki = 130 nM T40332 CSFN37 44309050 Ki = 0.39 nM T40332 CR4XO9 44309051 Ki = 1.1 nM T40332 CX80SC 44309073 Ki = 3.4 nM T40332 C18AZL 44309216 IC50 = 3.5 nM T40332 C8E0AZ 44309228 Ki = 15 nM T40332 CBEA34 44309326 Ki = 0.65 nM T40332 C60GWS 44312415 Ki > 100000 nM T40332 CDGX29 44312419 Ki = 3200 nM T40332 C75DJS 44312600 Ki > 100000 nM T40332 C9LT2C 44312642 IC50 = 20000 nM T40332 C61MLD 44312660 IC50 = 12000 nM T40332 CKHV96 44312681 IC50 = 3000 nM T40332 CK08ZX 44312691 IC50 = 9000 nM T40332 CIWU48 44312692 IC50 > 20000 nM T40332 CE06PC 44312711 IC50 = 800 nM T40332 C6HV5N 44312736 IC50 = 700 nM T40332 C6D8ZP 44312737 IC50 = 3000 nM T40332 CCBJ53 44312740 IC50 = 1000 nM T40332 C25UOL 44312741 IC50 = 2000 nM T40332 CB3A9W 44312771 IC50 > 20000 nM T40332 C1P7ED 44312773 IC50 = 3000 nM T40332 C4HJZ9 44312840 Ki = 4000 nM T40332 COYR46 44312861 Ki = 12000 nM T40332 C28YCZ 44312862 Ki = 400 nM T40332 C5GMQ9 44312896 Ki = 1500 nM T40332 C40UFA 44312925 IC50 > 20000 nM T40332 C37LOU 44312957 IC50 = 20000 nM T40332 CJQI56 44312958 IC50 = 4000 nM T40332 CQO41D 44312969 IC50 = 4000 nM T40332 C08ZBI 44312990 IC50 = 700 nM T40332 CU3E4B 44312991 IC50 = 100 nM T40332 CQJ5F9 44312992 IC50 = 4000 nM T40332 C2YA6T 44312993 Ki = 10000 nM T40332 CRZX02 44313005 IC50 = 2000 nM T40332 CCM2R1 44313033 IC50 = 2000 nM T40332 CT69SA 44313040 IC50 = 4000 nM T40332 CZ24YH 44313056 IC50 = 600 nM T40332 CG0Y5Z 44313064 IC50 = 700 nM T40332 CO01JG 44313077 IC50 = 300 nM T40332 CN1E5H 44313087 IC50 = 5000 nM T40332 C9LT4Z 44313114 IC50 = 4000 nM T40332 CJ5UI3 44313122 Ki = 50000 nM T40332 CC7A1J 44313131 Ki = 53000 nM T40332 C4UNO3 44313149 IC50 = 20000 nM T40332 CZ07MG 44313176 IC50 = 5000 nM T40332 C8VCL3 44313177 IC50 = 5000 nM T40332 CD2FS4 44313342 Ki = 22000 nM T40332 CQK72I 44313345 Ki = 1500 nM T40332 C2XHU4 44313650 Ki = 14000 nM T40332 CH18RW 44313833 Ki = 1300 nM T40332 CKN8C1 44316486 IC50 > 10000 nM T40332 C60AVB 44317117 Ki >= 30000 nM T40332 C4T0AC 44317137 Ki >= 88000 nM T40332 CCVZ83 44317149 Ki >= 72000 nM T40332 C83FQT 44317256 Ki = 43000 nM T40332 CP03CV 44317262 Ki >= 45000 nM T40332 CJ2B9M 44317267 Ki = 29000 nM T40332 C3T6YK 44317274 Ki >= 78000 nM T40332 C5AR9V 44317284 Ki >= 30000 nM T40332 CKP03R 44317285 Ki >= 104000 nM T40332 CAK4P6 44318572 IC50 = 40000 nM T40332 C84AGV 44319331 IC50 = 1400 nM T40332 C0CWH7 44319367 IC50 = 76000 nM T40332 C5Z8KW 44319375 IC50 = 43000 nM T40332 C1RL4T 44319383 IC50 = 45000 nM T40332 CO5CA2 44319384 IC50 = 94000 nM T40332 C3VH1X 44319419 IC50 = 13000 nM T40332 CAC49M 44319423 IC50 = 11000 nM T40332 C3GO1N 44319641 IC50 = 1600 nM T40332 CMPE25 44319642 IC50 = 18000 nM T40332 CM5HO4 44321916 Ki = 0.008 nM T40332 C4MJ8H 44322029 Ki = 0.01 nM T40332 CB3Q9U 44322389 Ki = 0.007 nM T40332 CA6KV2 44331082 Ki = 14.5 nM T40332 CBFS14 44331115 Ki = 2 nM T40332 CJ19RM 44337844 Ki = 0.64 nM T40332 C0TE6U 44337930 Ki = 0.64 nM T40332 CHT61Y 44338018 Ki = 8 nM T40332 C14UGI 44338019 Ki = 0.65 nM T40332 C0JY7C 44338029 Ki = 0.06 nM T40332 CWI7N9 44338415 IC50 = 5000 nM T40332 CN4C5X 44338416 IC50 = 5700 nM T40332 CZX39H 44338433 IC50 = 60 nM T40332 CXF5Z2 44338508 IC50 = 400 nM T40332 CBM7L9 44338509 IC50 = 3500 nM T40332 CU5H2I 44338658 IC50 = 900 nM T40332 CC0O3Q 44338659 IC50 = 220 nM T40332 C09SZK 44338660 IC50 = 450 nM T40332 C32EVN 44338707 IC50 = 1600 nM T40332 C06BSK 44338737 IC50 = 1400 nM T40332 CGM1H7 44338738 IC50 = 1800 nM T40332 C4XDT1 44338807 IC50 = 340 nM T40332 C6K3YE 44338808 IC50 = 900 nM T40332 CUFS02 44338809 IC50 = 560 nM T40332 CZD3L7 44338820 IC50 = 400 nM T40332 CMK10R 44338821 IC50 = 20 nM T40332 CP56NM 44338822 IC50 = 7300 nM T40332 CKP0B1 44339163 Ki = 34 nM T40332 CA1D5G 44339167 Ki = 1.6 nM T40332 C2FZD6 44339168 Ki = 51.6 nM T40332 C4HY8G 44339183 Ki > 100 nM T40332 C5R4DQ 44339184 Ki = 10 nM T40332 CPQ47M 44339196 Ki = 13.6 nM T40332 CEX5G4 44339197 Ki = 42 nM T40332 CG87DW 44339210 Ki > 1000 nM T40332 CWM73S 44339220 Ki > 100 nM T40332 C5JZA6 44340361 Ki = 1 nM T40332 C75HMC 44340504 Ki = 18 nM T40332 COE37X 44340528 Ki = 1 nM T40332 CE71WL 44340543 Ki = 5 nM T40332 CZE75W 44340561 Ki = 1 nM T40332 C54RWE 44340595 Ki = 100 nM T40332 CR4OT3 44341284 Ki = 1.1 nM T40332 C8J1KC 44341355 Ki = 2.2 nM T40332 C0XZO4 44341377 Ki = 0.2 nM T40332 CR8KP4 44341378 Ki = 5.2 nM T40332 CLQ2W9 44341406 Ki = 0.03 nM T40332 C2AT7J 44342409 Ki = 17 nM T40332 CUR86C 44342423 Ki = 20 nM T40332 CF60PZ 44342469 Ki = 1380 nM T40332 C8DV6S 44342778 IC50 = 9000000 nM T40332 CH3CE9 44342794 IC50 = 5400000 nM T40332 CWLT78 44342805 IC50 > 10000000 nM T40332 CWQ13J 44342806 IC50 > 10000000 nM T40332 CB7HO1 44342811 Ki = 4 nM T40332 C01YDQ 44342827 IC50 = 8900000 nM T40332 CX2HK7 44342836 IC50 > 10000000 nM T40332 C64PAR 44342837 IC50 = 2600000 nM T40332 CH39PO 44342847 IC50 > 10000000 nM T40332 CLI0B3 44342857 IC50 = 8900000 nM T40332 CP7RQ6 44342869 IC50 > 10000000 nM T40332 CJU1K9 44342887 IC50 = 2560000 nM T40332 CMR6I2 44342888 IC50 = 6410000 nM T40332 CXO27U 44342890 IC50 > 10000000 nM T40332 C95EXJ 44342891 IC50 = 210000 nM T40332 C9BKY1 44342937 IC50 = 5350000 nM T40332 CX6M5P 44342953 IC50 = 6000000 nM T40332 CN1VD4 44342954 IC50 = 1180000 nM T40332 CA93TW 44342991 IC50 = 490000 nM T40332 CBED26 44342992 IC50 > 10000000 nM T40332 CF0XD7 44343000 IC50 > 10000000 nM T40332 CTI5A0 44343012 IC50 = 2070000 nM T40332 C14ITM 44343019 IC50 = 13900000 nM T40332 CS8E1H 44343022 IC50 = 4270000 nM T40332 C9QD7A 44343029 IC50 = 6000000 nM T40332 COY26B 44343032 IC50 > 10000000 nM T40332 CKT05N 44343039 IC50 = 7100000 nM T40332 CNS1W4 44343061 IC50 = 6100000 nM T40332 C0JP1W 44343069 IC50 = 280000 nM T40332 C3KGY9 44343124 IC50 > 10000000 nM T40332 C4HFN2 44343139 IC50 = 3360000 nM T40332 CZT68I 44343164 IC50 = 390000 nM T40332 CJ6R9X 44343194 IC50 > 10000000 nM T40332 CQ7A9W 44343906 Ki > 100000 nM T40332 C9X0ZR 44343907 Ki > 100000 nM T40332 C6FY8O 44345532 IC50 = 12000 nM T40332 CPW75O 44348239 Ki = 250 nM T40332 C5U7YX 44348372 Ki = 500 nM T40332 CD8AL2 44351097 IC50 = 69 nM T40332 CHGE39 44351104 IC50 = 74 nM T40332 C2RMW4 44351162 IC50 = 88 nM T40332 C2Y7GN 44352045 Ki = 0.5 nM T40332 C68KSH 44352097 Ki = 1 nM T40332 C0D4CK 44353344 Ki = 1 nM T40332 C38RJF 44353357 Ki = 200 nM T40332 CQU69T 44353358 Ki = 7 nM T40332 COPM05 44353364 Ki = 66000 nM T40332 C20CYN 44353485 Ki < 0.1 nM T40332 CN85XQ 44354163 IC50 > 300000 nM T40332 CGL18R 44359861 Ki = 19 nM T40332 CLM3H4 44359870 Ki = 70 nM T40332 CL9GT7 44359932 Ki = 70 nM T40332 CD0PS5 44359934 Ki = 59 nM T40332 C80BKQ 44359984 Ki = 7 nM T40332 C9Z2IU 44359985 Ki = 2 nM T40332 C53AJT 44360051 Ki = 21 nM T40332 CY24NZ 44360093 Ki = 43 nM T40332 CJEC32 44360131 Ki = 44 nM T40332 CZ5JL3 44360132 Ki = 24 nM T40332 CIX34U 44360133 Ki = 39 nM T40332 C5NE7W 44360270 Ki = 29 nM T40332 CLO39R 44361701 Ki = 0.016 nM T40332 C1RS0F 44361716 Ki = 0.021 nM T40332 CO6VL0 44362002 Ki = 0.093 nM T40332 CHF49P 44362414 Ki = 120.23 nM T40332 CT04RY 44362423 Ki = 257.04 nM T40332 CAP5Y6 44362424 Ki = 102.33 nM T40332 C0W7TH 44362425 Ki = 14454.4 nM T40332 C93FWR 44362443 Ki = 0.0955 nM T40332 CKTI90 44362458 Ki = 1096.48 nM T40332 CGAN05 44362471 Ki = 12882.5 nM T40332 CHAQ14 44362472 Ki = 6918.31 nM T40332 C41XZU 44362486 Ki = 758.58 nM T40332 CSZ03H 44362546 Ki = 7585.78 nM T40332 CCHM90 44362570 Ki = 398.11 nM T40332 C2UZC3 44362571 Ki = 2570.4 nM T40332 C51UBY 44362573 Ki = 549.54 nM T40332 CLG37U 44362583 Ki = 363.08 nM T40332 C4FK2R 44362584 Ki = 70.79 nM T40332 C4XCT3 44362585 Ki = 467.74 nM T40332 C8O5YU 44362587 Ki = 104.71 nM T40332 CMK28R 44362631 Ki = 39.81 nM T40332 CT2X0F 44362640 Ki = 1548.82 nM T40332 CND9Z3 44362653 Ki = 1.585 nM T40332 C5XU6E 44362657 Ki = 181.97 nM T40332 CNEI94 44362661 Ki = 5100 nM T40332 C41HKG 44362664 Ki = 10 nM T40332 CH4YV7 44362667 Ki = 660.69 nM T40332 C7CR2Y 44362668 Ki = 741.31 nM T40332 C78ROB 44362669 Ki = 3388.44 nM T40332 C52GSX 44362683 Ki = 151.36 nM T40332 C7O9RC 44362688 Ki = 6456.54 nM T40332 C9U3FY 44362694 Ki = 97723.72 nM T40332 C2EIU0 44362697 Ki = 1122.02 nM T40332 C3Z6BO 44362707 Ki = 2137.96 nM T40332 CCDJ03 44362708 Ki = 109.65 nM T40332 CZ8BI0 44362721 Ki = 478.63 nM T40332 CO59RP 44362722 Ki = 338.84 nM T40332 C24FNJ 44362734 Ki = 169.82 nM T40332 CCD2N8 44362741 IC50 = 107 nM T40332 CLV72W 44362755 Ki = 1202.26 nM T40332 C4GRW1 44362756 Ki = 1445.44 nM T40332 CED8M4 44362761 Ki = 0.9333 nM T40332 C9YM0R 44362762 Ki = 72.44 nM T40332 C6N1FA 44362778 Ki = 1258.93 nM T40332 C8QFN6 44362779 Ki = 30.9 nM T40332 C0QG4Z 44362780 Ki = 537.03 nM T40332 CLI68E 44362789 Ki = 109.65 nM T40332 CNWF06 44362845 Ki = 8.128 nM T40332 CTAY98 44362846 Ki = 1.413 nM T40332 C06INC 44362848 Ki = 20.89 nM T40332 CY6QH7 44362849 Ki = 177.83 nM T40332 C6ZM5V 44362850 Ki = 114.82 nM T40332 C71WGV 44362853 Ki = 1230.27 nM T40332 CVH3L1 44362854 Ki = 1584.89 nM T40332 C2K7JM 44362855 Ki = 158489.32 nM T40332 C6P1AQ 44362869 Ki = 1698.24 nM T40332 CSEZ31 44362877 Ki = 446.68 nM T40332 C9FC7V 44362890 Ki = 1995.26 nM T40332 CKE47Z 44362891 Ki = 2137.96 nM T40332 CPL17T 44362892 Ki = 316.23 nM T40332 C67KRN 44362900 Ki = 724.44 nM T40332 CT0SE7 44362901 Ki = 239.88 nM T40332 CXZS62 44362903 Ki = 154.88 nM T40332 C3R8CM 44362909 Ki = 199.53 nM T40332 C6C8RO 44362910 Ki = 2.692 nM T40332 CK5AJ0 44362944 Ki = 28.18 nM T40332 CN43FB 44362945 Ki = 20.89 nM T40332 C2FRU6 44362954 Ki = 1000 nM T40332 CG48UP 44362959 Ki = 5495.41 nM T40332 C1ETU0 44362969 Ki = 39.81 nM T40332 CS3H1F 44362970 Ki = 7.762 nM T40332 CAO25V 44362980 IC50 = 365 nM T40332 CR8MD1 44362982 Ki = 72.44 nM T40332 CV4Z7R 44363005 Ki = 691.83 nM T40332 CPU7L1 44363006 Ki = 281.84 nM T40332 C72KXW 44363019 Ki = 21.38 nM T40332 CT7V2L 44363025 Ki = 54954.09 nM T40332 CUCE12 44363030 Ki = 21.38 nM T40332 C27SKX 44363034 Ki = 7943.28 nM T40332 CZK7I9 44363091 Ki = 65000 nM T40332 C7Q5UZ 44363092 Ki = 595000 nM T40332 CO6Z8K 44366639 Ki = 55 nM T40332 CFL1J0 44366665 Ki = 4 nM T40332 C27VSQ 44366666 Ki = 15.9 nM T40332 C35YGE 44367854 IC50 = 7800 nM T40332 C7FBC3 44367865 IC50 > 10000 nM T40332 CV4L8A 44367935 IC50 = 7.6 nM T40332 CD0IM7 44368008 IC50 = 8.9 nM T40332 C8E7CZ 44368051 IC50 = 130 nM T40332 CVM6S7 44368057 IC50 = 66 nM T40332 C9RLA3 44368068 IC50 > 10000 nM T40332 CR53IL 44368071 IC50 = 290 nM T40332 CU3F6L 44368072 IC50 = 230 nM T40332 C97NDU 44368076 IC50 > 10000 nM T40332 C4SFV3 44368077 IC50 > 10000 nM T40332 C5TQ1G 44368099 IC50 > 10000 nM T40332 C41CWE 44368121 IC50 > 10000 nM T40332 C1ZW4D 44368174 IC50 > 10000 nM T40332 C0BC2Q 44368175 IC50 > 10000 nM T40332 C6L9DK 44368178 IC50 = 450 nM T40332 CPE92K 44368218 IC50 = 7.2 nM T40332 C19ARS 44368431 IC50 > 10000 nM T40332 CMN18Z 44368433 IC50 = 13 nM T40332 C3S7YX 44368434 IC50 = 7.4 nM T40332 CIP7M3 44368435 IC50 > 10000 nM T40332 C62RSP 44368445 IC50 = 280 nM T40332 CV0Y2M 44368446 IC50 = 72 nM T40332 CCY58J 44368452 IC50 = 3.5 nM T40332 CSYO09 44368455 IC50 > 10000 nM T40332 CP6V1Y 44368456 IC50 > 10000 nM T40332 C0G6XP 44372603 Ki = 2 nM T40332 CQ6UZ3 44373218 IC50 > 5000 nM T40332 C0UE9N 44375714 IC50 = 0.365 ug.mL-1 T40332 CNFA42 44380213 IC50 = 380 nM T40332 CA84BI 44380230 IC50 = 74 nM T40332 CY5QC9 44380439 IC50 = 330 nM T40332 CD6AM9 44380440 IC50 = 320 nM T40332 CDMP49 44380948 Ki = 0.6 nM T40332 CVT80Q 44380960 Ki = 1.8 nM T40332 CED81F 44381178 Ki = 1.6 nM T40332 CKW3N0 44381293 Ki = 1.6 nM T40332 CO0X8N 44381295 Ki = 8000 nM T40332 CHI6Q5 44383146 IC50 = 26 nM T40332 C17LOX 44383308 IC50 = 274 nM T40332 CI3KG4 44383348 IC50 = 120 nM T40332 C0CW7E 44383468 IC50 = 242 nM T40332 CB3ED9 44383545 IC50 = 22 nM T40332 C1FCZ3 44384633 IC50 > 1000000 nM T40332 C8HL9B 44384637 IC50 = 810000 nM T40332 CR0T6A 44384638 IC50 = 665000 nM T40332 CTF25D 44384701 IC50 > 1000000 nM T40332 C2WSZ7 44384797 IC50 = 989000 nM T40332 CA0F5I 44384840 IC50 = 742000 nM T40332 CN0XD8 44384856 IC50 = 305000 nM T40332 CUBE67 44385436 IC50 = 454000 nM T40332 C8G1VT 44385622 IC50 = 92000 nM T40332 CLW2F7 44385646 IC50 = 895000 nM T40332 CF3GW6 44385689 IC50 > 1000000 nM T40332 C92XES 44385735 IC50 = 292000 nM T40332 CB35TE 44385740 IC50 > 1000000 nM T40332 C7W9MR 44385741 IC50 > 1000000 nM T40332 CU85DE 44385747 IC50 > 1000000 nM T40332 CK9I0A 44385748 IC50 > 1000000 nM T40332 CUAJ67 44385919 IC50 > 1000000 nM T40332 CJ98UI 44387451 IC50 = 41 nM T40332 C3JQH9 44398885 Ki = 2900 nM T40332 C0THI1 44415189 IC50 = 89800 nM T40332 CGDY32 44415219 IC50 = 75800 nM T40332 C6WR4P 44445934 Ki = 65 nM T40332 CA6E2R 44445935 Ki = 410 nM T40332 C3EBM1 44445936 Ki = 130 nM T40332 CBP7C3 44445937 Ki = 71 nM T40332 CE50KV 44452404 IC50 = 1560 nM T40332 C6M7VJ 44453668 Ki = 21000 nM T40332 C6J2PV 44453794 Ki = 6.4 nM T40332 CQT15C 44453896 Ki = 0.2 nM T40332 C2YA0P 44453914 Ki = 0.66 nM T40332 CUA0E6 44453915 Ki = 0.81 nM T40332 CN3K8S 44453963 Ki = 0.06 nM T40332 CMH91A 44454011 Ki = 0.35 nM T40332 CCP29L 44459365 Ki = 309 nM T40332 C20MDV 44459881 IC50 = 7000 nM T40332 CY34QH 44461452 Ki = 240 nM T40332 CSK2J8 44461627 Ki = 340 nM T40332 C5UHG2 44461629 Ki = 40 nM T40332 CU4O1C 44461630 Ki = 120 nM T40332 C7Y9HQ 44461644 Ki = 34 nM T40332 C82FIS 44461664 Ki = 9800 nM T40332 CG05CL 44461760 Ki = 400000 nM T40332 C23EAH 44461777 Ki = 20 nM T40332 C5RJ9A 44461780 Ki = 41000 nM T40332 C2R4ZM 44461781 Ki = 95000 nM T40332 CB0HR7 44461805 Ki = 1100 nM T40332 CZ4Q6H 44473061 IC50 = 7.6 nM T40332 C8WU0Y 44473063 IC50 = 43 nM T40332 CGA18I 44473064 IC50 = 42 nM T40332 CA8D5R 44473065 IC50 = 35 nM T40332 CCN52T 44473066 IC50 = 1000 nM T40332 CX4FB6 44473067 IC50 > 1000 nM T40332 C60FLK 44517752 IC50 = 8.1 nM T40332 CIT5G7 44561891 IC50 > 100000 nM T40332 C90BGR 44561892 IC50 > 100000 nM T40332 C9RGX4 44561893 IC50 > 100000 nM T40332 CU7NP5 44561930 IC50 > 100000 nM T40332 CV21IQ 44561931 IC50 = 33000 nM T40332 CR08WA 44561932 IC50 > 100000 nM T40332 C97JBD 44584781 IC50 > 100000 nM T40332 CBP4J9 44584783 IC50 > 100000 nM T40332 CUV18S 44584784 IC50 > 100000 nM T40332 C7ZYA5 44626812 Ki = 1.3 nM T40332 C98FOV 44626813 Ki = 33.9 nM T40332 CPG20K 44626906 Ki = 99.3 nM T40332 CJXK95 44626907 Ki = 7.6 nM T40332 CMXF01 44626997 Ki = 203 nM T40332 CR9I0Y 44626998 Ki = 0.82 nM T40332 COL76S 44626999 Ki = 0.34 nM T40332 CQS4G2 44627000 Ki = 1 nM T40332 C8KQH6 44627001 Ki = 1.1 nM T40332 C6V5XI 44627002 Ki = 0.5 nM T40332 CTP5R6 44627003 Ki = 1.8 nM T40332 CYO0Q2 44627268 IC50 = 16 nM T40332 C2PVE0 45103523 Ki > 26000 nM T40332 CGN14R 45103723 Ki > 26000 nM T40332 CJ0D8A 45267494 IC50 = 22 nM T40332 C32KHM 45267507 IC50 = 900 nM T40332 CY2VP7 45267519 IC50 = 8.6 nM T40332 CT18QR 45267524 IC50 = 28 nM T40332 CBS28A 45267536 IC50 = 850 nM T40332 CITF18 45268358 IC50 = 24 nM T40332 CKO71F 45268410 IC50 = 140 nM T40332 CL5GJ6 45268419 IC50 = 23 nM T40332 CLN7M0 45269246 IC50 = 79 nM T40332 C6K5CY 45269247 IC50 = 74 nM T40332 CKS94Q 45269257 IC50 = 5300 nM T40332 CSM9D3 45269258 IC50 = 2600 nM T40332 CIAG68 45269260 IC50 = 210 nM T40332 C90YKZ 45269266 IC50 = 15000 nM T40332 CM19HY 45269268 IC50 = 25 nM T40332 CPU0F3 45269270 IC50 = 28 nM T40332 C10DXZ 45270089 IC50 = 170 nM T40332 C6U2VN 45270092 IC50 = 160 nM T40332 COVE69 45270109 IC50 = 120 nM T40332 C6WZI7 45270119 IC50 = 27 nM T40332 CFY4G5 45270120 IC50 = 21 nM T40332 CMCK76 45270925 IC50 = 87 nM T40332 C5DC9K 45270953 IC50 = 150 nM T40332 CV1UK4 45271765 IC50 = 85 nM T40332 CAL64K 45271771 IC50 = 710 nM T40332 CLOK73 45271783 IC50 = 8.5 nM T40332 C8SM0J 45271784 IC50 = 20 nM T40332 CBW47X 45271792 IC50 = 330 nM T40332 C1BQ7N 45271797 IC50 = 34 nM T40332 C6SRB3 45272629 IC50 = 16 nM T40332 CND82I 45272646 IC50 = 28 nM T40332 C4U6MS 45272654 IC50 = 250 nM T40332 CTS68D 45272660 IC50 = 180 nM T40332 CES4L3 45273539 IC50 = 21 nM T40332 C5WYG0 45273548 IC50 = 9300 nM T40332 CYI53S 45273574 IC50 = 71 nM T40332 C5KYI2 45273582 IC50 = 140 nM T40332 CJ3MI1 45273583 IC50 = 110 nM T40332 C6T2AJ 45273590 IC50 = 1300 nM T40332 CD4T1L 46221636 Ki = 13000 nM T40332 CN7QI3 46221638 IC50 = 300 nM T40332 CF16UR 46225505 IC50 > 100000 nM T40332 C81XNC 46225794 IC50 = 33 nM T40332 C4YAJ7 46228924 IC50 > 10000 nM T40332 C46YMU 46838142 IC50 = 30.8 nM T40332 COP81J 46838143 IC50 = 30.7 nM T40332 C1PDI7 46838144 IC50 = 24.8 nM T40332 COQH23 46838145 IC50 = 48.8 nM T40332 CI19BN 46838146 IC50 = 15.4 nM T40332 CD28QR 46882316 Ki > 7500 nM T40332 C86FZA 46882318 Ki = 32 nM T40332 C3G9BA 46882319 Ki = 21 nM T40332 C8JFN6 46882328 Ki = 520 nM T40332 CUI91D 46905615 IC50 = 1900 nM T40332 CX8S3H 46933351 Ki = 7340 nM T40332 C41UEJ 49759015 IC50 = 2400 nM T40332 CJH50R 49797481 IC50 > 100000 nM T40332 CI7P2B 49797571 IC50 = 170 nM T40332 CI59MV 49797572 IC50 > 30000 nM T40332 C96CKU 49797573 IC50 = 220 nM T40332 C50QVP 53262865 IC50 = 830 nM T40332 C6AFX0 53320723 IC50 = 500 nM T40332 CCR6H5 53357861 IC50 = 89 nM T40332 CI9GP5 53357862 IC50 = 130 nM T40332 C52ZET 53357863 IC50 = 240 nM T40332 C53JUT 53357864 IC50 = 260 nM T40332 C9YK0S 53357865 IC50 = 180 nM T40332 CP7ZW2 53784885 IC50 = 0.036 nM T40332 CBJQ98 54132077 IC50 = 370 nM T40332 C0WH1K 54675757 Ki = 8128305.16 nM T40332 CNEI60 54678950 Ki = 1100000 nM T40332 CL42YZ 54685126 Ki = 93325.43 nM T40332 C29BYX 54686804 Ki = 1700000 nM T40332 CJ6BS7 54690337 Ki = 6309573.44 nM T40332 CPQ05N 54693753 IC50 = 3150000 nM T40332 CY4VG6 54693756 IC50 = 1620000 nM T40332 CQ85OF 54694046 Ki = 4897788.19 nM T40332 CV0U6E 54694048 Ki = 10000000 nM T40332 C95DEC 54694049 Ki = 645654.23 nM T40332 C9FGL4 54694052 Ki = 6025595.86 nM T40332 C01LMD 54694053 Ki = 489778.82 nM T40332 C1K4RP 54695445 IC50 = 26800 nM T40332 CL4N6C 54707146 Ki = 95499.26 nM T40332 C9FQ0U 54709932 IC50 = 35800 nM T40332 C5FPG9 54728809 IC50 = 153000 nM T40332 C28IAV 54732424 Ki = 151356.12 nM T40332 C1T9XJ 54733673 Ki = 977237.22 nM T40332 COA25T 54733674 Ki = 363078.05 nM T40332 CJ4LH1 54735926 Ki = 400000 nM T40332 CPGD29 56598201 IC50 = 9280 nM T40332 C6QCK2 56598333 IC50 > 20000 nM T40332 C8U4OD 56649692 IC50 > 1000000 nM T40332 C8QC6E 56659686 IC50 = 29000 nM T40332 CFTW24 56659687 IC50 = 5900 nM T40332 C6TDH1 56659688 IC50 = 8100 nM T40332 C4A7XT 56659690 IC50 = 36000 nM T40332 C2Y7HM 56659691 IC50 = 930 nM T40332 C3LO5F 56659692 IC50 = 1600 nM T40332 CJ0AU4 56659693 IC50 = 400 nM T40332 C0FP7U 56659694 IC50 = 780 nM T40332 CZ1RB3 56659695 IC50 = 650 nM T40332 C9C6SF 56659699 IC50 = 22000 nM T40332 C8GT6J 56663146 IC50 = 3900 nM T40332 CX8BK7 56663147 IC50 = 6100 nM T40332 CVEQ14 56663148 IC50 = 11000 nM T40332 C0A9JD 56663149 IC50 = 52000 nM T40332 CZS51B 56663151 IC50 = 310 nM T40332 CA9LH5 56663152 IC50 = 1900 nM T40332 CFL20B 56663153 IC50 = 510 nM T40332 CAXE63 56663154 IC50 = 890 nM T40332 CM7DT1 56663155 IC50 = 510 nM T40332 CS3O6Z 56663156 IC50 = 340 nM T40332 C9HUK8 56666600 IC50 = 38000 nM T40332 C1CV4T 56666601 IC50 = 25000 nM T40332 CJPL65 56666602 IC50 = 410 nM T40332 C7RWF1 56666605 IC50 = 700 nM T40332 C12FWP 56666606 IC50 = 690 nM T40332 CWH4G9 56666607 IC50 = 480 nM T40332 CVU62F 56670016 IC50 = 1800 nM T40332 C4GJH8 56670017 IC50 = 3100 nM T40332 CFMA80 56670019 IC50 = 10000 nM T40332 CL20GF 56673430 IC50 = 800 nM T40332 CDH38Y 56673525 IC50 = 33000 nM T40332 C7ET5S 56673526 IC50 = 1700 nM T40332 CY4JH2 56673529 IC50 = 550 nM T40332 C1MN5G 56673530 IC50 = 400 nM T40332 C3TUR8 56674980 Ki = 269700 nM T40332 CY5R9M 56676773 IC50 = 420 nM T40332 CSC9U1 56676774 IC50 = 34000 nM T40332 CK9YG2 56676775 IC50 = 930 nM T40332 C5P4NQ 56676842 IC50 = 1700 nM T40332 C8NC2F 56676843 IC50 = 38000 nM T40332 C74KYG 56676844 IC50 = 460 nM T40332 C0AV1L 56680166 IC50 = 3100 nM T40332 CY1TH5 56680168 IC50 = 28000 nM T40332 C4SW5X 56680170 IC50 = 1900 nM T40332 CAJN07 56683509 IC50 = 760 nM T40332 C0UIF5 57671050 IC50 > 100000 nM T40332 CY26NE 57671116 IC50 > 10000 nM T40332 C9E6CB 57671131 IC50 > 10000 nM T40332 CJO75X 57671161 IC50 > 10000 nM T40332 CTH9W2 58343687 IC50 = 2700 nM T40332 CDZ05M 59145670 IC50 = 3.5 nM T40332 C5ON3H 60195210 IC50 = 680 nM T40332 C48UHX 66561877 IC50 = 2600 nM T40332 CL93DE 66725365 IC50 = 17 nM T40332 C17JAZ 68284084 IC50 > 30000 nM T40332 CTP6M3 70681508 IC50 > 500000 nM T40332 C25DHK 70685488 IC50 >> 5000 nM T40332 CD9N4J 70687893 IC50 > 500000 nM T40332 CLW0V4 70687894 IC50 > 500000 nM T40332 C3SZ6M 70696249 IC50 > 500000 nM T40332 C8JPF6 71450320 Ki = 5000 nM T40332 C06BIJ 71452128 Ki = 4000 nM T40332 CBU34G 71452812 IC50 = 7000 nM T40332 C03DMT 71452813 IC50 = 15000 nM T40332 CKG69H 71454592 IC50 = 700 nM T40332 C0XV2L 71455698 IC50 = 14000 nM T40332 CH8C9Z 71455699 IC50 > 200000 nM T40332 C6TI5U 71455700 IC50 > 200000 nM T40332 C3A8KU 71456312 IC50 = 3000 nM T40332 CL62BK 71457475 IC50 = 300 nM T40332 CF9XP4 71457476 IC50 > 200000 nM T40332 C96SGY 71457477 IC50 = 46000 nM T40332 CU9O8L 71459588 Ki = 0.6 nM T40332 CZH4E8 71460024 IC50 = 600 nM T40332 CF5O8M 71461119 IC50 = 39000 nM T40332 CH87QX 71461740 IC50 = 300 nM T40332 C2PKD0 71462857 IC50 = 51000 nM T40332 C83ZNH 71562308 IC50 = 40 nM T40332 CL9VA2 71562455 IC50 = 121 nM T40332 CTJR81 71562563 IC50 = 28 nM T40332 C6LB5N 71659627 IC50 = 8400 nM T40332 C0DPM1 71659628 IC50 > 100000 nM T40332 CRH4J2 71659766 IC50 > 100000 nM T40332 C2BDV0 71659767 IC50 = 46600 nM T40332 C78DJQ 71711730 IC50 < 10000 nM T40332 C51TZR 71717105 IC50 = 21 nM T40332 CQIA07 71717727 IC50 = 195 nM T40332 CULQ46 71718935 IC50 = 41 nM T40332 CL23VT 71723878 IC50 > 100000 nM T40332 C5RSD4 71818404 IC50 = 20 nM T40332 CS0OQ1 71818406 IC50 = 330 nM T40332 CXO32I 71818543 IC50 = 310 nM T40332 CDH81R 71818544 IC50 = 140 nM T40332 COX58Z 71818547 IC50 = 31 nM T40332 CQ9OD7 71818548 IC50 = 40 nM T40332 CVPL10 71818549 IC50 = 7 nM T40332 C6X9AY 71818550 IC50 = 260 nM T40332 CKS7E3 71818686 IC50 = 12500 nM T40332 CY7ZS9 71818687 IC50 = 6400 nM T40332 CVCM38 71818688 IC50 = 30 nM T40332 CA56TS 71818689 IC50 = 15 nM T40332 C1S2VT 71818690 IC50 = 50 nM T40332 CFV7P5 71818691 IC50 = 50 nM T40332 CK2XH0 71818692 IC50 = 20 nM T40332 CXV8Z4 71818829 IC50 = 25 nM T40332 C7UY4N 71818830 IC50 = 30 nM T40332 C6X2FC 71818831 IC50 = 30 nM T40332 C80YBP 71818832 IC50 = 18 nM T40332 CKCP90 71818833 IC50 = 50 nM T40332 CYC57T 71818834 IC50 = 210 nM T40332 C2D1NZ 71818963 IC50 = 100 nM T40332 CXV20J 71818964 IC50 = 12 nM T40332 C2M1ZG 71818965 IC50 = 50 nM T40332 CLV3J9 71818966 IC50 = 330 nM T40332 CQI96C 71819101 IC50 = 80 nM T40332 CY82VQ 71819102 IC50 = 80 nM T40332 CL3KA5 71819103 IC50 = 210 nM T40332 CWY8D4 71819104 IC50 = 160 nM T40332 CQ1K8Y 71819105 IC50 = 80 nM T40332 C2NP3X 71819106 IC50 = 270 nM T40332 CL8I3R 71819107 IC50 = 260 nM T40332 C4QL2M 71819248 IC50 = 220 nM T40332 C7HQD3 71819249 IC50 = 150 nM T40332 CSDL97 71819250 IC50 = 100 nM T40332 CYF8I9 71819251 IC50 = 80 nM T40332 CCKZ58 71819252 IC50 = 140 nM T40332 CMXU14 71819253 IC50 = 60 nM T40332 CO72XA 71819254 IC50 = 110 nM T40332 CR43YH 71819387 IC50 = 6400 nM T40332 CW3QR2 72712049 Ki = 68700 nM T40332 CAL2W7 72712050 Ki = 11300 nM T40332 C2A4TH 72712051 Ki > 250000 nM T40332 CN73TI 72712053 Ki > 250000 nM T40332 C3J8RV 72712070 Ki > 250000 nM T40332 C8QJ2R 72793725 IC50 = 450 nM T40332 CG9R4L 72793726 IC50 = 4100 nM T40332 CHLW60 72793743 IC50 = 8900 nM T40332 C7J9MS 72793744 IC50 = 14300 nM T40332 CC28PB 72793745 IC50 > 50000 nM T40332 C60WDY 72793746 IC50 = 670 nM T40332 C1MBU7 72793747 IC50 = 110 nM T40332 CBT72J 72793748 IC50 = 1190 nM T40332 CP7XG2 72793760 IC50 = 1200 nM T40332 CETY07 72793761 IC50 = 4600 nM T40332 CNF72C 72793762 IC50 = 5190 nM T40332 C76CUL 72793763 IC50 = 960 nM T40332 C9MWN6 72793764 IC50 = 300 nM T40332 CLY96J 72793765 IC50 = 280 nM T40332 C6BY5D 72793776 IC50 = 180 nM T40332 CHL95X 72793777 IC50 = 2460 nM T40332 C1DI8A 72793778 IC50 = 80 nM T40332 CNU1I7 73051428 IC50 < 20 nM T40332 C10ITF 73345210 IC50 >> 5000 nM T40332 CR7HX5 73345258 IC50 = 2 nM T40332 C4E7TG 73345260 IC50 = 94 nM T40332 C7BKZ5 73345448 IC50 = 100 nM T40332 CR3E1A 73345466 Ki = 17 nM T40332 C14AZB 73345741 Ki = 3.9 nM T40332 C3M6NT 73345742 Ki = 15 nM T40332 CV0TP1 73345743 Ki = 150 nM T40332 C5KHS8 73347173 Ki = 1200 nM T40332 CD26JR 73347227 Ki = 7.8 nM T40332 C04QVO 73347230 IC50 = 32 nM T40332 C5AMR2 73348056 IC50 = 7800 nM T40332 CL1Z5W 73348476 Ki = 500 nM T40332 C8OMT5 73348493 Ki = 43 nM T40332 CTP68V 73348565 Ki = 200 nM T40332 CE26GR 73348743 Ki = 2 nM T40332 C4XN1F 73348744 Ki = 0.63 nM T40332 CD6HY8 73349819 IC50 >> 5000 nM T40332 C87PWL 73349864 IC50 = 31 nM T40332 C0ONC3 73350318 Ki = 2.9 nM T40332 CU0H6E 73350319 Ki = 14 nM T40332 CH4L7K 73350322 IC50 = 210 nM T40332 CO01PD 73351555 IC50 = 30 nM T40332 CRQS78 73351639 Ki = 44 nM T40332 CXL3Q6 73351830 Ki = 16 nM T40332 C8TOM4 73351831 Ki = 0.96 nM T40332 CH52ZV 73351832 Ki = 3.8 nM T40332 CVGO29 73352827 IC50 = 29 nM T40332 C7BYL1 73353012 IC50 = 120000 nM T40332 C84NFB 73353013 IC50 = 60 nM T40332 C8TC2M 73353039 Ki = 1.9 nM T40332 CKSD62 73353041 Ki = 20 nM T40332 COQ9E0 73353305 Ki = 2.6 nM T40332 CTWH20 73353306 Ki = 45 nM T40332 C2CM8U 73354616 Ki = 234.42 nM T40332 C4DVG0 73354687 Ki = 210 nM T40332 CO3A5T 73354820 Ki = 1 nM T40332 C48MTS 73354821 Ki = 11 nM T40332 C3OTL1 73355884 IC50 = 172 nM T40332 C04GZD 73355907 IC50 = 0.69 nM T40332 CY81IS 73356107 IC50 > 1000000 nM T40332 C84MDZ 73356367 Ki = 6.8 nM T40332 CS15MB 73356368 Ki = 810 nM T40332 CJ2DF3 73356369 Ki = 20 nM T40332 CX17VC 76284943 IC50 < 20 nM T40332 CALM86 76335198 Ki = 0.4 nM T40332 CP6T1S 77844774 IC50 = 22 nM T40332 CAL1Y8 77844829 IC50 < 1 nM T40332 CGM61S 77844945 IC50 < 1 nM T40332 CH7GQ9 86268083 IC50 = 74700 nM T40332 C53SOM 90310890 IC50 = 2.4 nM T40332 CM06KI 90311037 IC50 = 1.6 nM T40332 CP50TI 90643774 Ki = 38000 nM T40332 CG2Q3B 90643775 Ki = 22000 nM T40332 CJKX87 90643776 Ki = 36000 nM T40332 CU9WA6 90643777 Ki = 39000 nM T40332 CK89GM 90643778 Ki = 39000 nM T40332 CF0R9S 90643779 Ki = 39000 nM T40332 CU5N9Z 90663487 IC50 = 107 nM T40332 CH1OE8 90666510 IC50 > 100000 nM T40332 C7ZCN4 90676239 IC50 = 4400 nM T40332 C6IO0L 90676242 IC50 = 1400 nM T40332 C4S9WP 90676243 IC50 = 900 nM T40332 C8O4GH 90676244 IC50 > 10000 nM T40332 C0CTE9 90676245 IC50 = 500 nM T40332 C7GDE8 90676248 IC50 = 500 nM T40332 C25ZWA 90676249 IC50 = 1100 nM T40332 C7OX2A 90676250 IC50 = 2900 nM T40332 CMV0H1 90676258 IC50 = 1500 nM T40332 C8E4WS 102323332 IC50 > 50000 nM T40332 CR2AU7 118010068 IC50 = 320 nM T40332 COA36C 118010069 IC50 = 370 nM T40332 C5NJH1 118202505 IC50 = 680 nM T40332 C43ADS 118202506 IC50 = 110 nM T40332 C2UXT7 118202507 IC50 = 50 nM T40332 CPV27G 118202509 IC50 = 120 nM T40332 CJB3K7 118202510 IC50 = 190 nM T40332 C12BHL 118202511 IC50 = 360 nM T40332 COT6H0 118202512 IC50 = 370 nM T40332 CFS4A9 118716662 IC50 = 3.7 nM T40332 C2WNT9 118716663 EC50 < 1 nM T40332 C8ZSC2 118727248 IC50 = 2240 nM T40332 CYIX41 118727249 IC50 = 390 nM T40332 CH1T3M 118727250 IC50 = 820 nM T40332 CVG1X5 118727251 IC50 = 480 nM T40332 C9B6KX 118727252 IC50 = 1230 nM T40332 C3OUW6 118727253 IC50 > 10000 nM T40332 C10QJC 118727254 IC50 > 10000 nM T40332 CVIF56 118727255 IC50 > 10000 nM T40332 CNQ9U4 118727256 IC50 = 3690 nM T40332 CN93WU 118727257 IC50 > 10000 nM T40332 C5DR7Z 118727258 IC50 > 10000 nM T40332 CDEU05 118727259 IC50 = 130 nM T40332 CZHT12 118727260 IC50 = 290 nM T40332 C3WC9Y 121488127 IC50 > 100000 nM T40332 CKJN32 122164799 IC50 > 30000 nM T40332 CYEA84 122190691 IC50 < 1 nM T40332 C9QKI3 127020966 IC50 > 100000 nM T40332 CE26HW 131955087 IC50 > 100000 nM T40332 CES7P6 132517499 IC50 = 21000 nM T40332 CGE51P 135672692 IC50 = 2910 nM T40332 C7YVL9 135981708 IC50 = 3010 nM T40332 CZ9X0E 137634272 IC50 = 51900 nM T40332 CNL2Z9 137635679 Ki = 12000 nM T40332 C43ETF 137637257 IC50 = 47600 nM T40332 C7BQ8O 137644210 IC50 = 19100 nM T40332 C9BEA1 137644608 IC50 = 64800 nM T40332 C6BE7C 137646856 IC50 = 157000 nM T40332 C03IMN 137647139 Ki = 8900 nM T40332 CNO2T8 137647340 IC50 = 230 nM T40332 CME1B3 137649275 IC50 = 810 nM T40332 C7WRB2 137652193 IC50 = 640 nM T40332 CZ1H4R 137655362 Ki = 43000 nM T40332 C47IZA 137655464 IC50 = 1560 nM T40332 CVN59W 137656193 IC50 = 91300 nM T40332 C34UDN 137657165 IC50 = 2650 nM T40332 C0C5JK 137657334 IC50 = 320 nM T40332 CTUM82 137658421 IC50 = 690 nM T40332 CUZ35A 138115400 IC50 > 100000 nM T40332 C6OP2I 140742745 IC50 = 250 nM T40332 CZT48W 140742746 IC50 = 7000 nM T40332 C61ODQ 145952347 Ki = 3200 nM T40332 C10EWY 145953439 IC50 > 100000 nM T40332 C5WFZ3 145955487 Ki = 6300 nM T40332 C1ZYD7 145955680 Ki = 12400 nM T40332 CFOI32 145956166 Ki = 19500 nM T40332 C1MJ0P 145957172 IC50 = 2400 nM T40332 C95HXU 145958432 IC50 = 35600 nM T40332 C27FNP 145960559 Ki = 13100 nM T40332 C9OK4P 145979023 IC50 = 800 nM T40332 C0CJ8N 145979295 IC50 = 12600 nM T40332 C2KTP8 145979350 IC50 = 1500 nM T40332 CZ2S6U 145979786 IC50 = 80 nM T40332 CLYZ05 145980145 IC50 = 6700 nM T40332 CWBN57 145980442 IC50 = 490 nM T40332 CCT8O7 145980848 IC50 = 7300 nM T40332 C6B2NR 145981285 IC50 = 11900 nM T40332 CVE50X 145982102 IC50 = 44800 nM T40332 CDT82U 145982407 IC50 = 87 nM T40332 CSL8R0 145985380 IC50 = 640 nM T40332 CJW50C 145986748 IC50 = 3400 nM T40332 CS0V3Y 145987313 IC50 = 19100 nM T40332 CO1PC5 145987373 IC50 = 15 nM T40332 CI5AZ8 145987496 IC50 = 2600 nM T40332 CNHI09 145988102 IC50 = 1500 nM T40332 CCD6J8 145988308 IC50 = 28500 nM T40332 C9EJT1 145988325 IC50 = 38500 nM T40332 CW2HO0 145988348 IC50 = 42600 nM T40332 CR8V9N 145988581 IC50 = 3600 nM T40332 C8PIN1 145988987 IC50 = 1800 nM T40332 CD6ZT8 145989305 IC50 = 24 nM T40332 CM1G6B 145989653 IC50 = 6000 nM T40332 CJT4G6 145990495 IC50 = 11500 nM T40332 C0XQV5 145990804 IC50 = 620 nM T40332 CT7R5S 145990987 IC50 = 14 nM T40332 CCJF05 145991040 IC50 = 1800 nM T40332 C91SQO 145991281 IC50 = 2400 nM T40332 CDW8L7 145991384 IC50 = 770 nM T40332 CHZ5V0 145993786 IC50 = 390 nM T40332 CSBC71 146680900 IC50 = 55000 nM T40332 CH82XM 155511283 IC50 = 4710 nM T40332 CZR36C 155511554 IC50 = 12589.25 nM T40332 CSL60M 155511684 IC50 = 3230 nM T40332 CT3GQ1 155517665 IC50 = 197 nM T40332 C9HK4E 155519617 IC50 = 1540 nM T40332 C6NX4K 155519661 IC50 > 100000 nM T40332 C4MS1B 155519676 IC50 = 100000 nM T40332 C7L5RK 155520356 IC50 = 103 nM T40332 CH1Y5O 155522603 IC50 = 10100 nM T40332 C9KE6J 155524006 IC50 = 2190 nM T40332 CBU5W0 155524880 Ki = 24 nM T40332 CN3BH5 155527998 IC50 = 794.33 nM T40332 CL4RC9 155528080 IC50 = 595 nM T40332 CHYW65 155528639 IC50 = 1258.93 nM T40332 CLJI15 155529200 IC50 = 2350 nM T40332 CD7O2G 155530095 IC50 = 31622.78 nM T40332 C3W2MJ 155530593 IC50 = 35800 nM T40332 C35QWO 155531023 IC50 > 100000 nM T40332 C2X5EJ 155531124 IC50 > 10000 nM T40332 C50ZHO 155533944 IC50 = 4830 nM T40332 CJB82P 155535066 IC50 = 5850 nM T40332 C10QDI 155535871 IC50 = 2600 nM T40332 C12HON 155536142 IC50 > 100000 nM T40332 CHUF10 155537107 IC50 > 500000 nM T40332 CX6S5M 155537400 IC50 = 140 nM T40332 CZMX52 155540843 IC50 = 10000 nM T40332 CY6DK3 155540964 IC50 = 15848.93 nM T40332 CG8OY6 155543393 IC50 = 1350 nM T40332 CV9N7I 155543726 IC50 = 21700 nM T40332 C5MB9R 155547962 IC50 = 6309.57 nM T40332 CLFB25 155548371 IC50 = 25118.86 nM T40332 CS57LN 155549377 IC50 = 2340 nM T40332 CUF2J6 155550172 IC50 = 840 nM T40332 CWC8X9 155550748 IC50 > 100000 nM T40332 COM52R 155551892 IC50 = 1584.89 nM T40332 CJ3FI5 155553630 IC50 > 100000 nM T40332 C2E5GR 155554478 Ki = 3.2 nM T40332 CJL26S 155555493 IC50 = 400 nM T40332 CE3G5W 155556110 IC50 > 10000 nM T40332 C0SND3 155557259 IC50 > 10000 nM T40332 C7E2NJ 155557306 IC50 > 10000 nM T40332 CA38JF 155557625 IC50 = 360 nM T40332 CSW48V 155557718 IC50 > 100000 nM T40332 CTS63Q 155558248 IC50 > 10000 nM T40332 CFX07G 155558369 Ki = 16 nM T40332 C9X7TF 155560751 IC50 = 450 nM T40332 C6JPU5 155564831 IC50 = 6300 nM T40332 CM8XB1 155565537 IC50 = 5011.87 nM T40332 CS54OQ 155566050 IC50 = 680 nM T40332 CW96TS 155566656 IC50 > 150000 nM T40332 CU42CE 155567829 IC50 > 100000 nM T40332 CQA3R5 155569370 IC50 = 721 nM T40332 CY9GR5 10009357 IC50 = 11100 nM T40332 CAI36L 10101940 IC50 = 404 nM T40332 C4BL1N 10327685 IC50 = 69 nM T40332 C7OHD3 10350525 IC50 = 4900 nM T40332 CAUB96 10440265 IC50 = 57 nM T40332 CX6PI4 14861876 IC50 = 153 nM T40332 CF4B3J 21832914 IC50 = 65 nM T40332 C4PVG3 44372915 IC50 = 138 nM T40332 CR1T4Y 44372920 IC50 = 5100 nM T40332 CJ8ZU5 44372983 IC50 > 5000 nM T40332 C4T1XJ 44372984 IC50 = 1562 nM T40332 CNLX57 44373015 IC50 > 5000 nM T40332 CT7R5D 44373019 IC50 = 30 nM T40332 CGX5Q3 44373020 IC50 = 84 nM T40332 C6KD9P 44373025 IC50 = 73 nM T40332 C9ZSG2 44373051 IC50 = 693 nM T40332 C18WIL 44373075 IC50 = 817 nM T40332 C0W3BJ 44373137 IC50 > 5000 nM T40332 CEN6O7 44373154 IC50 = 57 nM T40332 CO1H7G 44373162 IC50 = 149 nM T40332 CQOI69 44373163 IC50 = 175 nM T40332 CE7W2Y 44373173 IC50 > 5000 nM T40332 C23GOW 44373196 IC50 > 5000 nM T40332 C3DX2N 44373204 IC50 = 110 nM T40332 CPL8V3 44373205 IC50 = 52 nM T40332 CUI13J 44373211 IC50 = 452 nM T40332 CY0Z5O 44373212 IC50 = 5000 nM T40332 C1JMP8 44373240 IC50 = 61 nM T40332 C91JLZ 44373268 IC50 = 73 nM T40332 CYK80J 44373269 IC50 = 92 nM T40332 CJP5G2 44373315 IC50 = 156 nM T40332 CK78NM 44373333 IC50 = 153 nM T40332 CEK35P 44373526 IC50 = 217 nM T40332 C8DQ4W 44373542 IC50 = 507 nM T40332 C2N0KC 44373543 IC50 = 67 nM T40332 C8CJ2N 9986046 IC50 > 5000 nM T40332 CLNZ94 9986475 IC50 = 635 nM T40332 C68QAJ 9988180 IC50 > 5000 nM T40332 D00RIX 5280443 IC50 = 46100 nM T40332 D00TYW 54678949 Ki = 15000 nM T40332 D00WFQ 674641 Ki = 65 nM T40332 D02AKP 695069 Ki = 2500 nM T40332 D02AVL 18376720 Ki > 5000 nM T40332 D02NRY 674650 Ki = 300 nM T40332 D02PAU 16731825 Ki = 10000 nM T40332 D03BNM 10053241 Ki = 3 nM T40332 D03MNO 121963 Ki = 2.2 nM T40332 D03STO 24823606 Ki = 114 nM T40332 D04KAS 44454029 Ki = 73 nM T40332 D04ODG 44626814 Ki = 3.9 nM T40332 D04SPO 44584782 IC50 = 18000 nM T40332 D05ICF 3492365 IC50 = 230 nM T40332 D05ZIP 674656 Ki = 45 nM T40332 D06GTS 76318115 IC50 = 630 nM T40332 D06JMS 44626902 Ki = 4450 nM T40332 D06LPR 674651 Ki = 34 nM T40332 D07DOW 685230 Ki = 3400 nM T40332 D07HLC 24823444 Ki = 34.4 nM T40332 D07IBU 10696098 IC50 > 10000 nM T40332 D08OCS 699665 Ki = 28 nM T40332 D08RPN 674653 Ki = 250 nM T40332 D08WQJ 700133 Ki = 46 nM T40332 D09FGQ 123985 IC50 > 300000 nM T40332 D0A5ZF 44626811 Ki = 2.2 nM T40332 D0B4WZ 44626901 Ki = 127 nM T40332 D0C1NP 66561876 IC50 = 10200 nM T40332 D0D6ZB 25205741 IC50 = 7 nM T40332 D0E0EQ 708205 Ki = 110 nM T40332 D0F2YC 10038543 IC50 = 100 nM T40332 D0F3CA 1609 IC50 = 100 nM T40332 D0H8EO 139973 Ki = 1.21 nM T40332 D0I1AC 577102 Ki = 230 nM T40332 D0IU5E 716930 Ki = 39 nM T40332 D0J1LX 24882417 IC50 = 540 nM T40332 D0L8DL 9889727 Ki = 0.27 nM T40332 D0MQ8A 20283207 Ki = 0.85 nM T40332 D0N9DP 54737457 Ki = 4600 nM T40332 D0O8PM 669334 Ki = 290 nM T40332 D0PQ8B 54736658 Ki = 7900 nM T40332 D0Q7ST 44338671 IC50 = 800 nM T40332 D0R9CH 3400921 Ki > 10000 nM T40332 D0S5RY 4784 IC50 = 52161.7 nM T40332 D0T9WZ 54613196 IC50 = 4220 nM T40332 D0X1OY 674628 Ki = 104 nM T40332 D0Z7LS 44626810 Ki = 233 nM T16691 D00KHM 16362 Ki = 71 nM T16691 D01AZG 5073 Ki = 224 nM T16691 D01XBA 5035 Ki = 750 nM T16691 D01ZII 2726 Ki = 4 nM T16691 D03WEX 9966051 Ki = 330 nM T16691 D04JEE 4946 EC50 > 5011.87 nM T16691 D04VFJ 3005573 Ki = 4125 nM T16691 D04WFD 4543 Ki = 214 nM T16691 D06YFA 31101 Ki < 50 nM T16691 D07KSG 2733526 Ki = 1041 nM T16691 D08VRO 3822 Ki = 2800 nM T16691 D0B0CP 667467 Ki = 3 nM T16691 D0CQ0Z 33630 Ki = 1000 nM T16691 D0D1AL 3559 Ki = 1083 nM T16691 D0G8NN 119570 Ki > 10000 nM T16691 D0H3HM 60795 Ki = 89 nM T16691 D0H7KF 5002 Ki > 1000 nM T16691 D0I8LU 5311507 Ki = 169 nM T16691 D0MA9N 2955 Ki = 183 nM T16691 D0P5SA 3372 Ki < 50 nM T16691 D0R1JV 60854 Ki = 20 nM T16691 D0R6RO 4184 Ki = 55 nM T16691 D0U5FS 3396 Ki = 1188 nM T16691 D0U5OE 3964 Ki = 15 nM T16691 D0V4QS 135398745 Ki = 5 nM T16691 D0W5HK 216239 Ki = 6213 nM T16691 D0Z1RV 135398737 Ki = 4 nM T16691 D0ZS8P 2801 Ki = 112 nM T16691 D08CJK 1150 Ki = 70 nM T16691 D09IRN 21071390 Ki = 0.83 nM T16691 D0N1HW 5311200 Ki = 1656.2 nM T16691 D0R9HI 11256720 Ki = 0.166 nM T16691 D0V4ZQ 16071605 Ki = 1.3 nM T16691 D00OWF 5280953 Ki = 1480 nM T16691 D02JMI 9888211 Ki = 398.11 nM T16691 D03PJW 108029 IC50 = 79 nM T16691 D06DZI 107780 Ki > 10000 nM T16691 D06ZVC 10150497 Ki = 2 nM T16691 D08AWI 11430856 Ki > 5000 nM T16691 D0B7SP 11292933 Ki > 5011.87 nM T16691 D0M7LV 5761 Ki = 6.31 nM T16691 D0OS6O 60149 Ki = 5 nM T16691 D0Q2JS 10436045 Ki = 79.43 nM T16691 D0YP7L 6604889 Ki = 6309.57 nM T16691 C36WOC 2800 Ki = 1956 nM T16691 CJ0B9F 3158 Ki = 105 nM T16691 C5H9CN 9287 Ki = 909 nM T16691 C2TYP0 31386 Ki = 1598 nM T16691 C6WDL7 49756 Ki = 60 nM T16691 CTB26S 52899 Ki = 80 nM T16691 C3PWO1 77956 Ki = 491 nM T16691 C0ALO6 152215 Ki = 98 nM T16691 CGT8R0 160510 Ki = 1450 nM T16691 CLK7P3 169713 IC50 = 16 nM T16691 CLG13W 227584 Ki = 482 nM T16691 C5BNW8 235964 Ki = 630.96 nM T16691 CYV1R3 417052 Ki = 1930 nM T16691 CN2RL6 460659 Ki = 564 nM T16691 CYZ25A 563919 Ki = 10 nM T16691 C1EY3K 616691 Ki = 33 nM T16691 CKR2N7 621659 IC50 = 370 nM T16691 CLUH96 627240 Ki = 114 nM T16691 C86DOU 640912 Ki = 866 nM T16691 C1QWJ9 675366 Ki = 198 nM T16691 CXQ6U0 735755 IC50 > 10000 nM T16691 C1RC8P 744368 Ki > 5000 nM T16691 C2VLP8 752521 Ki = 696 nM T16691 CXB86D 846090 Ki = 875 nM T16691 C6N9QC 1244725 Ki = 61 nM T16691 C9FI5L 1296368 Ki = 15610 nM T16691 C08VKR 1472656 Ki = 237 nM T16691 C6VZT7 1984087 Ki = 2700 nM T16691 CGS9R7 2133793 Ki = 7886 nM T16691 CG9N3A 2136365 Ki = 1174 nM T16691 CT8KN9 2232766 Ki = 2539 nM T16691 CA2OY6 2737389 Ki = 596 nM T16691 CBK16O 2771410 Ki = 28 nM T16691 C0QTF4 2771418 Ki = 482 nM T16691 CP8NQ2 2771419 Ki = 25 nM T16691 CP9O0G 2771422 Ki = 1512 nM T16691 CPI2C5 2775690 Ki = 1262 nM T16691 C29YXF 2816054 Ki = 5700 nM T16691 C1C4LH 2843443 Ki = 12730 nM T16691 CO4MP2 2845118 Ki = 250 nM T16691 C7UVI2 2848343 Ki = 1221 nM T16691 CRA6F5 2853434 Ki = 3104 nM T16691 CB6EK5 2854567 Ki = 80 nM T16691 C41ULI 2855326 Ki = 245 nM T16691 C6DL8S 2866185 Ki = 1490 nM T16691 C3QRD6 2867758 Ki = 5800 nM T16691 C9WY0K 2870667 Ki = 8 nM T16691 CL2G3H 2870750 Ki = 6401 nM T16691 CC74QS 2872937 Ki = 9669 nM T16691 C2G4DQ 2876391 Ki = 5 nM T16691 CRF65H 2880253 Ki = 5600 nM T16691 C54SFI 2883218 Ki = 894 nM T16691 C6L8FJ 2891368 Ki = 119 nM T16691 C7KJ4R 2894562 Ki = 290 nM T16691 CH4X1C 2906325 Ki = 12 nM T16691 CFE09S 2906372 Ki = 1267 nM T16691 CT4VY7 2906559 Ki = 61 nM T16691 CET7C8 2921525 Ki = 3700 nM T16691 C2DE6R 2927683 Ki = 1400 nM T16691 CF01YE 2928642 Ki = 2500 nM T16691 CY8R6Q 2948971 Ki = 670 nM T16691 CLXQ01 2950739 Ki = 2400 nM T16691 CO0C7J 2962174 Ki = 1900 nM T16691 C1U5AG 3028929 Ki = 6.5 nM T16691 C5F4AI 3028955 Ki = 12 nM T16691 CAM8H3 3066250 IC50 = 80 nM T16691 C6SA2G 3132842 Ki = 3400 nM T16691 C2W7DI 3142696 Ki = 163 nM T16691 CNX8I1 3245407 EC50 = 1100 nM T16691 CEG3M8 3643745 Ki = 26 nM T16691 CS8KE2 3649661 Ki = 3587 nM T16691 CKN8W0 3950432 Ki = 20 nM T16691 CRC1M5 4494260 Ki = 59 nM T16691 C6SHA4 4713248 Ki = 2600 nM T16691 CRUB15 4723431 Ki = 91 nM T16691 C9H5AV 4723679 Ki = 266 nM T16691 CSL48K 4725280 Ki = 185 nM T16691 CZ64GQ 4976400 Ki = 774 nM T16691 C7N1KM 5206725 Ki = 4489 nM T16691 C4J3HP 5640104 Ki = 5676 nM T16691 C35XAN 6484477 Ki = 316 nM T16691 C1O2PM 6625986 IC50 = 5000 nM T16691 C0QCK1 6918455 Ki = 1.259 nM T16691 CU3X9A 6918479 Ki = 0.85 nM T16691 CN5LJ4 6918531 Ki = 50 nM T16691 CW0ZE5 6918542 Ki = 2 nM T16691 CE6GX4 6918576 Ki = 25.12 nM T16691 C5V0WQ 6918577 Ki = 1.995 nM T16691 CW8OV4 6918578 Ki = 1.259 nM T16691 CEP3W2 6918579 Ki = 1.585 nM T16691 CC5PQ0 6918601 Ki = 7.2 nM T16691 C1WXY3 6918603 Ki = 1.995 nM T16691 C5GJ8Z 6918629 Ki = 1.4 nM T16691 CD0Z4I 6918648 Ki = 0.6 nM T16691 C2EJL3 6918682 Ki = 0.5 nM T16691 C8AL9V 6918689 Ki = 1 nM T16691 C0Y9VE 6918715 Ki = 0.2 nM T16691 C02GXO 6918745 Ki = 0.1259 nM T16691 CCLE83 6918748 Ki = 29 nM T16691 CI5L3H 6918751 Ki = 0.2 nM T16691 CH9GT8 6918786 Ki = 0.04 nM T16691 C2F3BY 7125890 Ki = 1574 nM T16691 CH57FQ 7183407 IC50 = 860 nM T16691 CV57DN 7184883 Ki = 2.8 nM T16691 CPX40Y 7184886 Ki = 30.2 nM T16691 CN2Z0K 7184892 IC50 = 580 nM T16691 CAV70B 7184895 IC50 = 1490 nM T16691 CG7B6O 7184976 IC50 = 1570 nM T16691 C81PDS 7185121 IC50 = 69 nM T16691 C2MGC8 7185122 IC50 = 190 nM T16691 C13EFJ 7185123 Ki = 3.2 nM T16691 CG09XB 7185124 Ki = 87.5 nM T16691 C6CDV7 7185128 IC50 = 1200 nM T16691 CD8UQ0 7246142 IC50 = 470 nM T16691 C57ZPS 7470702 IC50 = 1900 nM T16691 CUD06Z 9796627 Ki = 54 nM T16691 CFC9Y5 9799318 Ki < 1000 nM T16691 CV6PK5 9799635 Ki = 12 nM T16691 CR8GU7 9800707 Ki = 3.1 nM T16691 CL4QT6 9802776 Ki = 0.6 nM T16691 CB8Q2P 9803937 Ki = 3.162 nM T16691 CE0DI5 9804612 Ki < 6309.57 nM T16691 C89KNW 9805455 Ki = 2.512 nM T16691 CNX4F0 9805456 Ki = 1.259 nM T16691 CWOS30 9817810 Ki = 2.4 nM T16691 CPJA40 9817950 Ki = 370 nM T16691 C3BK4L 9821904 Ki = 11 nM T16691 C1JSL5 9822215 Ki = 1.5 nM T16691 CA5ID3 9822810 Ki = 0.3 nM T16691 C41ELD 9824783 Ki = 3 nM T16691 CM4I1N 9825329 Ki = 3.981 nM T16691 CR9H2E 9827562 Ki = 7.943 nM T16691 CNA93Z 9840981 Ki = 0.3 nM T16691 C4QVD7 9841077 Ki = 19 nM T16691 CTLV76 9841434 Ki = 3.8 nM T16691 C21IJU 9842551 Ki = 1 nM T16691 CI96TG 9847669 Ki = 1.995 nM T16691 CEM28L 9849116 Ki = 6.31 nM T16691 CM13ZV 9856041 Ki = 400 nM T16691 C0ZR3E 9861687 IC50 > 10000 nM T16691 CNCK78 9862256 Ki = 1.5 nM T16691 CO5YD2 9863380 Ki = 33 nM T16691 C0Q6AD 9863611 Ki = 1.995 nM T16691 C6Z9MV 9863836 Ki = 1.4 nM T16691 C9WBO2 9865474 Ki = 5.7 nM T16691 C0WBI8 9866222 Ki = 4.9 nM T16691 CG3NI8 9867263 Ki = 1.259 nM T16691 CB1F0C 9867475 Ki = 3 nM T16691 C7AB8O 9870053 Ki = 1.259 nM T16691 C2MKO6 9885426 Ki = 8.3 nM T16691 C08DBF 9885982 Ki = 4066 nM T16691 CJW1P5 9888494 Ki < 5011.87 nM T16691 C6N8UE 9889681 Ki = 0.5012 nM T16691 CM52WU 9890119 Ki = 1 nM T16691 CEG1K5 9891002 Ki = 1 nM T16691 C7QMK5 9891617 Ki = 1.259 nM T16691 CEL29O 9891618 Ki = 1 nM T16691 C3J8GU 9892409 Ki = 5.012 nM T16691 C7CD9N 9903598 Ki = 1030 nM T16691 CHFP46 9903970 Ki = 0.25 nM T16691 C9X1IV 9905247 Ki = 18 nM T16691 CUN81Q 9905249 Ki > 10000 nM T16691 C7NPZ0 9906059 Ki = 7.9 nM T16691 CYWQ50 9906447 Ki > 10000 nM T16691 CRK69H 9907512 Ki = 45 nM T16691 CAI90C 9908552 Ki = 7.9 nM T16691 CYZ5N4 9909089 Ki > 10000 nM T16691 CR52JI 9910619 Ki = 0.2 nM T16691 C9B3EA 9911844 Ki < 1000 nM T16691 C78MDV 9913554 Ki = 0.7943 nM T16691 C1IE8Y 9914461 Ki = 19.95 nM T16691 CR9KM0 9921064 IC50 = 40 nM T16691 CZQD80 9923440 Ki = 9 nM T16691 CA7RU6 9924293 Ki = 2.7 nM T16691 CMO2Y8 9924959 Ki = 2 nM T16691 C4UYZ7 9927441 Ki = 2.9 nM T16691 CV6A1D 9929294 Ki = 5 nM T16691 C9E1UB 9929665 Ki = 3.7 nM T16691 CTF52Q 9931929 Ki = 1 nM T16691 CGQ1A6 9933223 Ki = 1.7 nM T16691 CYVZ47 9934284 Ki < 1000 nM T16691 CWO45F 9935387 Ki = 0.7943 nM T16691 C6D7SX 9935750 Ki = 1.585 nM T16691 CGBP91 9945214 Ki = 58 nM T16691 CYH3R7 9947817 Ki = 1120 nM T16691 CQG0P3 9949258 Ki = 143 nM T16691 C67MTC 9950255 Ki = 0.3 nM T16691 CDKP85 9950402 Ki = 2 nM T16691 CDU68J 9952250 Ki = 8 nM T16691 CSBZ98 9953284 Ki = 1.6 nM T16691 CK8NR2 9954121 Ki = 0.631 nM T16691 CHOJ30 9956365 Ki < 1000 nM T16691 C96YVG 9956634 Ki = 0.3 nM T16691 CFR41N 9957068 Ki < 10000 nM T16691 C2CO7R 9957092 Ki = 1.995 nM T16691 CGR57X 9969402 IC50 = 7.3 nM T16691 CK9DF0 9976690 IC50 = 8.8 nM T16691 CFN50J 9978683 Ki = 1.6 nM T16691 C86FOH 9979009 Ki = 6 nM T16691 CFZ97V 9979313 Ki = 113 nM T16691 CWPT83 9979611 Ki = 0.7079 nM T16691 CRW7U6 9979748 IC50 = 12 nM T16691 C2T1WG 9983033 Ki = 27.6 nM T16691 CVOD42 9998950 IC50 = 28 nM T16691 C4BS8G 9999118 Ki = 7.3 nM T16691 CN3D2U 10019089 Ki = 0.2 nM T16691 CV7R9F 10020040 Ki > 10000 nM T16691 CU6Q5L 10020454 IC50 = 3.4 nM T16691 CK18LT 10020895 Ki > 10000 nM T16691 C8WTP3 10021389 IC50 = 70.1 nM T16691 C40IDM 10023874 Ki = 4.3 nM T16691 CB8VQ5 10024749 Ki = 15.5 nM T16691 CR9LM8 10026658 Ki = 2.13 nM T16691 CH59BP 10027190 Ki = 0.3 nM T16691 CD4J7G 10027518 Ki = 17 nM T16691 C2EUY0 10035109 Ki > 10000 nM T16691 C57TZR 10042333 Ki > 10000 nM T16691 COH3W5 10047631 Ki = 1.3 nM T16691 C8Z6MA 10067306 Ki = 2.3 nM T16691 CIK38G 10068007 Ki = 5.2 nM T16691 CD7T2M 10069527 Ki = 25.1 nM T16691 C6L3NU 10069592 Ki = 2.3 nM T16691 CV16DZ 10088284 Ki = 141 nM T16691 CZ5Y6U 10090742 IC50 = 83 nM T16691 COC0K5 10091305 IC50 = 57 nM T16691 CB0TU4 10091389 Ki = 9.6 nM T16691 C1XH8C 10091613 Ki = 8.76 nM T16691 CXF8S6 10091667 Ki = 20 nM T16691 C1SXF3 10094169 Ki = 18.3 nM T16691 CA3YF7 10094519 IC50 = 60 nM T16691 C63MGZ 10111488 Ki = 350 nM T16691 CT2X0H 10112809 Ki = 4.7 nM T16691 CJE70W 10112810 Ki = 0.4 nM T16691 CK2OR3 10112811 Ki = 4.3 nM T16691 CFO2L3 10113751 Ki = 5.3 nM T16691 C7G4BL 10113852 Ki = 163.5 nM T16691 C3NJ8W 10115005 Ki = 3 nM T16691 C8LD2B 10115854 Ki = 1 nM T16691 CXW68C 10117854 Ki = 9 nM T16691 CIB71R 10131565 Ki = 40 nM T16691 C36BMN 10134086 Ki = 0.3162 nM T16691 C0N8OY 10136185 Ki = 3 nM T16691 C2LS7U 10136837 Ki = 1 nM T16691 CQP7C9 10140915 Ki = 15 nM T16691 CAE3I7 10141477 Ki = 14 nM T16691 CET4Q9 10149997 Ki = 25.12 nM T16691 CC8RH3 10156341 Ki = 0.3981 nM T16691 CD6Y2A 10156556 Ki = 1.259 nM T16691 CCKZ54 10156876 Ki = 44 nM T16691 C7TL2R 10157412 Ki = 0.8 nM T16691 CSI1E5 10158456 Ki = 24.3 nM T16691 CT4FQ0 10159058 Ki = 4.5 nM T16691 C0GPO6 10162467 Ki = 1 nM T16691 C2J8TV 10172764 Ki = 0.34 nM T16691 CP6Q1W 10173403 Ki = 5.012 nM T16691 C2L8PI 10177503 Ki = 1.585 nM T16691 CB61DW 10177537 Ki = 7 nM T16691 CK6X9V 10178788 Ki = 0.5 nM T16691 C2AJ4U 10180527 Ki = 3.5 nM T16691 CUB5O8 10182052 Ki = 44 nM T16691 C1NLY7 10182109 Ki = 3.162 nM T16691 CQG3N5 10182228 Ki = 1 nM T16691 CFIB73 10182243 Ki = 0.1 nM T16691 CT7Q4V 10199220 Ki = 620 nM T16691 CWD43X 10199819 Ki = 3 nM T16691 CV4A2P 10201610 Ki = 1 nM T16691 C6W0YL 10202396 Ki = 5.3 nM T16691 C16DXL 10202995 Ki = 8 nM T16691 CV7S0G 10203339 Ki = 132 nM T16691 C1ET9N 10203612 Ki = 9.3 nM T16691 CW7EI0 10205655 Ki = 4 nM T16691 CFJY39 10216820 Ki = 5.012 nM T16691 CV1B7C 10217687 Ki = 10 nM T16691 CZ0TL1 10228179 Ki = 15.1 nM T16691 CI4W8Z 10246185 IC50 = 52 nM T16691 C6VO9Y 10246789 Ki = 18 nM T16691 CX85KT 10246904 IC50 = 42 nM T16691 CUHR59 10247229 IC50 = 87.6 nM T16691 CLT62K 10249280 IC50 = 68.9 nM T16691 C7MT4V 10250472 Ki = 0.6 nM T16691 CR96OK 10252130 Ki = 122 nM T16691 CSPF93 10252272 Ki = 3.981 nM T16691 CMRA02 10257042 Ki = 1995.26 nM T16691 CH31DX 10267394 Ki > 10000 nM T16691 CLG1B8 10269916 Ki = 63 nM T16691 C0T3SA 10270799 Ki = 2 nM T16691 CWV06I 10270854 Ki = 0.2512 nM T16691 CS3XW9 10272325 Ki = 5 nM T16691 CGU4I1 10272846 Ki = 10 nM T16691 C2D4BU 10273087 Ki = 1.995 nM T16691 C93SJA 10274389 Ki = 1 nM T16691 C85XYH 10275386 Ki = 6.8 nM T16691 CWQ21X 10276057 Ki = 3.3 nM T16691 C23PDE 10278839 Ki = 0.5 nM T16691 CA31LF 10286330 Ki = 1.995 nM T16691 CO2LT5 10286610 Ki = 3.981 nM T16691 C83QPR 10291754 Ki = 1 nM T16691 C7HP9C 10293741 Ki = 2.512 nM T16691 C51EXQ 10295001 Ki = 6.31 nM T16691 CAD92Z 10295665 Ki = 21.2 nM T16691 CR37BF 10296699 Ki = 163 nM T16691 CA3SK2 10297610 Ki = 3.9 nM T16691 CU89JD 10314060 Ki = 7385 nM T16691 CFQ54B 10315621 Ki = 98 nM T16691 C9U0DZ 10319296 Ki = 0.9 nM T16691 CHS1W3 10320800 Ki = 1.995 nM T16691 C04XAL 10341241 IC50 = 60 nM T16691 C8S4EN 10342674 Ki = 49 nM T16691 C9IAV3 10346043 Ki = 1 nM T16691 C4IL7N 10362440 IC50 = 79.2 nM T16691 CY8UH2 10364512 IC50 = 420 nM T16691 CR3KU9 10380133 Ki = 5.5 nM T16691 CMZA83 10383646 Ki = 1.9 nM T16691 C2P7OJ 10383682 IC50 = 0.7 nM T16691 CFAO13 10385670 IC50 = 470 nM T16691 C8L1IC 10390318 Ki = 10.3 nM T16691 CI1RB4 10405986 Ki = 3.2 nM T16691 C04WGF 10407367 Ki = 1 nM T16691 C5Y1TN 10409272 IC50 = 56 nM T16691 C4TPN1 10413595 Ki = 0.3162 nM T16691 C07AHG 10427672 IC50 = 1.3 nM T16691 CRMB96 10427673 IC50 = 41 nM T16691 C45CAU 10427896 IC50 = 22 nM T16691 CR4LS0 10430623 Ki = 1.1 nM T16691 CD7U5I 10433930 Ki = 1.995 nM T16691 CFLA92 10449488 Ki = 1 nM T16691 C3TF6V 10450930 Ki = 96 nM T16691 CN2WK7 10451504 IC50 = 11 nM T16691 C6H7GP 10452816 IC50 = 65 nM T16691 CL5J1E 10465905 Ki > 1000 nM T16691 CQD86O 10470893 IC50 = 2.4 nM T16691 COV85C 10472143 Ki = 15 nM T16691 C5LBS7 10472158 Ki = 2 nM T16691 C1UC7T 10472756 IC50 = 120 nM T16691 C26KCR 10475231 Ki > 1000 nM T16691 CEF2O6 10478367 Ki = 2410 nM T16691 C6XSG7 10480841 Ki = 200 nM T16691 CO0HE1 10498813 Ki = 10 nM T16691 CL70NJ 10499156 Ki < 10000 nM T16691 CQ4Y0V 10500364 Ki = 63.1 nM T16691 C85LRB 10505579 Ki = 1 nM T16691 CKAO03 10526615 Ki = 1.995 nM T16691 C3VLB5 10528182 Ki = 1.259 nM T16691 C75ZKM 10541285 Ki = 1258.93 nM T16691 C04EWM 10563312 Ki = 185 nM T16691 CHE80N 10573876 Ki = 3162.28 nM T16691 CN85DJ 10637020 Ki = 63.1 nM T16691 CP1UH5 10648664 Ki = 0.7943 nM T16691 CLE8P2 10658135 Ki = 24.3 nM T16691 CBRZ19 10658892 Ki = 168 nM T16691 C1Y3ON 10708918 Ki = 1000 nM T16691 C7XUR8 10713238 Ki = 20 nM T16691 C0V4PY 10757046 Ki = 200 nM T16691 C58CSG 10769116 Ki = 3.162 nM T16691 C3VTG2 10777767 Ki = 200 nM T16691 CJNM19 10800458 Ki = 240 nM T16691 CF34UD 10808841 Ki = 794.33 nM T16691 C0PE1N 10811310 Ki = 79.43 nM T16691 CD62XF 10825266 Ki = 130 nM T16691 CF3N5R 10826203 IC50 = 2 nM T16691 CNZ17B 10837078 Ki = 0.7943 nM T16691 CVT7J1 10873805 Ki = 300 nM T16691 CRI50E 10885636 IC50 = 2280 nM T16691 CX65PW 10907460 IC50 = 800 nM T16691 CNB39C 10947658 Ki = 13 nM T16691 C51NOQ 10982183 Ki ~ 0.1 nM T16691 CK6VF7 10991109 Ki = 3000 nM T16691 C4O7MD 10994400 Ki = 430 nM T16691 CM2R5C 11003533 Ki = 130 nM T16691 CJC9K4 11005810 IC50 = 427 nM T16691 C63DAE 11014674 Ki = 50.12 nM T16691 C3FIP5 11016205 Ki = 138 nM T16691 CS0Z2D 11024311 Ki = 2.291 nM T16691 CC05LI 11064294 Ki = 19.95 nM T16691 CG41BK 11071079 IC50 = 1530 nM T16691 C5AZ0I 11079889 Ki = 1700 nM T16691 C7DE0U 11113605 IC50 = 1350 nM T16691 CVE8T3 11121216 Ki = 61 nM T16691 COA02J 11154032 Ki = 9 nM T16691 CB1MG4 11154465 Ki = 1.9 nM T16691 CWS6J2 11162301 IC50 = 3580 nM T16691 CW7Y9O 11163741 Ki = 25.12 nM T16691 CX0YB7 11164580 Ki = 1 nM T16691 C8ZN3B 11166042 IC50 > 10000 nM T16691 CZ4C8S 11166043 Ki = 100.8 nM T16691 C1YA7F 11166261 Ki = 125.8 nM T16691 CV7PC9 11176859 Ki = 19.8 nM T16691 CA3Q8R 11177383 Ki = 3 nM T16691 C5U0JK 11177658 Ki = 116.2 nM T16691 C6CL1Y 11178830 Ki < 10000 nM T16691 C7YWQ1 11190151 Ki = 50.12 nM T16691 CCI40B 11190716 Ki > 1000 nM T16691 C17ZJO 11200157 EC50 = 5.2 nM T16691 C9N5QU 11200511 Ki = 1 nM T16691 C5YT1X 11200890 Ki = 0.631 nM T16691 CG7IR2 11201712 Ki > 1000 nM T16691 CPDU74 11201726 IC50 = 1.6 nM T16691 CAN97Q 11210467 EC50 = 1.4 nM T16691 C7ESF4 11210523 Ki > 1000 nM T16691 C94AIS 11211722 Ki = 1 nM T16691 C6D1MZ 11223004 EC50 = 1.3 nM T16691 CR04PZ 11232643 Ki = 4500 nM T16691 CD9XA5 11234629 EC50 = 0.8 nM T16691 C5XGC0 11234781 Ki = 57.7 nM T16691 CZE1A5 11235953 Ki = 10 nM T16691 COE13K 11236269 Ki = 9.8 nM T16691 CC4RT3 11237275 Ki > 1000 nM T16691 C1E0SQ 11245641 Ki = 4 nM T16691 CE97VF 11246907 Ki = 1 nM T16691 C90WSG 11248705 Ki < 10000 nM T16691 CBUP32 11257897 Ki = 41.2 nM T16691 CQ90VJ 11258709 Ki = 74.5 nM T16691 CZD6N4 11259180 Ki = 74.6 nM T16691 CI84OD 11259419 Ki = 90.2 nM T16691 CGJK46 11259456 Ki > 1000 nM T16691 CAU5P1 11260183 Ki = 1 nM T16691 C2VKI7 11269402 Ki = 64.7 nM T16691 CJNT47 11270131 Ki = 140.5 nM T16691 C7G8HX 11270546 Ki = 165.9 nM T16691 CQZE84 11271219 Ki = 31.4 nM T16691 CW7A0S 11280663 Ki = 1 nM T16691 C4JTQ3 11280771 Ki = 131 nM T16691 CM54IK 11282295 Ki = 194.8 nM T16691 C9HYZ8 11282389 Ki = 18.4 nM T16691 CTH8D9 11282884 IC50 = 1.1 nM T16691 CNZ23G 11283016 Ki = 224.4 nM T16691 CDRV20 11294169 Ki > 1000 nM T16691 C9BLC7 11304596 Ki = 3162.28 nM T16691 CJS9C0 11304851 IC50 > 7900 nM T16691 C30MTX 11306131 Ki = 336 nM T16691 CI79LV 11307899 Ki = 50.12 nM T16691 CZ0RP8 11314681 Ki = 1 nM T16691 C8Y7ZH 11316095 Ki = 1 nM T16691 CV6D3C 11316536 Ki = 12 nM T16691 CC9TE2 11316594 EC50 = 4.2 nM T16691 C46YHW 11316967 Ki = 9.6 nM T16691 C4Y5FE 11317551 Ki = 7.2 nM T16691 CW67JC 11326086 Ki = 0.9 nM T16691 CQ81DR 11328408 Ki > 1000 nM T16691 CL7QR0 11333554 EC50 = 130 nM T16691 CR89ME 11338273 Ki = 36 nM T16691 C42HTF 11338378 Ki = 14.9 nM T16691 CF6D5Z 11350253 Ki = 5.7 nM T16691 C1QKY2 11351089 Ki = 0.4 nM T16691 CGD42N 11361090 IC50 = 0.4 nM T16691 CWO59Z 11362134 Ki = 18.6 nM T16691 CY27GK 11363934 Ki = 0.3 nM T16691 CHB4E1 11371056 Ki = 1.2 nM T16691 C9QTU4 11372111 Ki = 16 nM T16691 CKF72Y 11383202 Ki = 4 nM T16691 C76EVG 11383990 Ki = 34 nM T16691 CBV52J 11384146 Ki = 0.4 nM T16691 CR46IF 11384675 Ki = 51.7 nM T16691 CX54VZ 11384694 Ki = 151.9 nM T16691 C1W7MS 11385064 Ki = 1 nM T16691 CJ74CP 11396708 IC50 = 0.8 nM T16691 CF4OX6 11397149 Ki = 316.23 nM T16691 C7MD9R 11406161 Ki = 4 nM T16691 CQ87XW 11407072 Ki = 0.3162 nM T16691 CM7I9Q 11407151 Ki = 85.8 nM T16691 CBV7Q8 11407544 Ki = 35 nM T16691 CK0FG2 11407867 Ki = 3 nM T16691 C1AYG7 11408932 Ki = 107.4 nM T16691 CR49LD 11408954 Ki > 1000 nM T16691 CK1A9Y 11417978 Ki = 94.2 nM T16691 C4X7AS 11418830 Ki = 3 nM T16691 CHV83P 11419238 Ki = 1 nM T16691 CB51AS 11420098 Ki = 108.8 nM T16691 C0FP4Z 11429601 Ki = 22 nM T16691 C85LYP 11430418 IC50 > 1000 nM T16691 CDWV48 11430512 Ki = 246.2 nM T16691 C6KHG1 11440676 Ki = 3 nM T16691 CY9B8H 11441064 Ki = 11 nM T16691 CV84SK 11441983 Ki = 7 nM T16691 C0L5RN 11442097 Ki = 124.5 nM T16691 C16DOF 11451904 Ki = 1 nM T16691 C6AF5E 11452988 Ki = 4 nM T16691 COH39T 11453792 Ki = 1 nM T16691 CD5FG4 11463428 EC50 = 1 nM T16691 CE7JU3 11463924 Ki = 123.6 nM T16691 CG75FW 11464995 Ki = 131.3 nM T16691 C24SNG 11474995 Ki = 1 nM T16691 CPS97N 11475760 Ki = 55.2 nM T16691 C59GHW 11476019 Ki = 24 nM T16691 CYJQ37 11476494 Ki = 97.3 nM T16691 CO6N3B 11486933 Ki = 1 nM T16691 CIWO57 11501251 Ki = 462 nM T16691 CO97GC 11501432 Ki = 346 nM T16691 CJK63T 11503175 Ki = 0.7943 nM T16691 CLU4R7 11504338 Ki > 1000 nM T16691 CIFQ02 11508173 Ki = 715 nM T16691 C7YD0A 11515129 Ki = 728 nM T16691 CD8I9H 11515192 Ki = 0.3162 nM T16691 CHK79E 11522477 Ki = 409 nM T16691 C6O9PM 11522698 Ki = 1013 nM T16691 C70RAX 11524473 IC50 = 0.8 nM T16691 CG0D5S 11532574 Ki = 4 nM T16691 CY4R9L 11545169 Ki = 3.6 nM T16691 C1V5CH 11559090 Ki = 30.1 nM T16691 CGP56Q 11559141 Ki = 164 nM T16691 CT1DE9 11560362 Ki = 304 nM T16691 C4TI1E 11566597 Ki = 0.4 nM T16691 CJ9UY6 11566775 Ki > 1000 nM T16691 CEM42D 11567716 Ki = 196.9 nM T16691 C25RSU 11567840 Ki = 77.5 nM T16691 CK3F1Y 11569025 Ki = 0.3 nM T16691 CO58PR 11573559 Ki = 156 nM T16691 CE23IV 11574113 Ki = 28.3 nM T16691 CBW12V 11574663 Ki = 9.2 nM T16691 C8NMI4 11575479 Ki = 82.4 nM T16691 C6D1MA 11584660 Ki > 1258.93 nM T16691 CN21IG 11587610 Ki = 0.3 nM T16691 C1M2CP 11589069 Ki = 580 nM T16691 CU45DK 11595209 Ki = 12.3 nM T16691 CV9B8R 11595360 Ki = 0.1585 nM T16691 CGX8F6 11596869 Ki > 1790000 nM T16691 C21XTO 11601657 Ki > 1000 nM T16691 CVQ4R6 11601955 Ki = 108 nM T16691 CN2F6O 11603453 Ki = 928 nM T16691 COY20C 11609368 Ki = 344.6 nM T16691 C4J6KG 11616729 Ki > 1000 nM T16691 C6V3OY 11624561 Ki = 0.3 nM T16691 CCK08F 11630209 Ki > 1000 nM T16691 CK6U7Q 11630824 Ki = 481 nM T16691 CHS76B 11631738 Ki = 877 nM T16691 CCY41R 11631819 Ki = 0.4 nM T16691 COH4T9 11632439 Ki = 19 nM T16691 COL12H 11638206 Ki = 27 nM T16691 C2OU7Y 11638332 Ki = 54.7 nM T16691 CD84ZC 11639865 Ki = 0.1995 nM T16691 CJ8ZS6 11640142 Ki > 1000 nM T16691 CV49QH 11652654 Ki = 0.2 nM T16691 C1HDM5 11653679 Ki = 295.9 nM T16691 C3KMW6 11653799 Ki > 1000 nM T16691 C5YC4N 11654089 Ki > 1000 nM T16691 C9X6PO 11661320 Ki = 1284 nM T16691 CE0C3N 11667340 Ki = 172 nM T16691 CRKQ54 11674694 Ki = 147 nM T16691 C8BNM7 11681803 Ki = 257 nM T16691 CRU61B 11682024 Ki = 0.3162 nM T16691 CB95CX 11683768 Ki = 952 nM T16691 CML4E8 11688736 Ki = 0.631 nM T16691 CZM75X 11689373 Ki = 1.259 nM T16691 C93ACF 11695841 Ki = 59 nM T16691 C23VNU 11697242 Ki = 0.3981 nM T16691 C2Q6TW 11703226 Ki = 73.2 nM T16691 C4G1EZ 11709684 Ki = 23 nM T16691 CG87CL 11716331 Ki = 1365 nM T16691 CV69CM 11723168 Ki = 3 nM T16691 CC37TI 11724023 IC50 = 2 nM T16691 C0NH2T 11724112 IC50 = 12 nM T16691 CP0QV2 11725253 IC50 = 250 nM T16691 CQA4Y1 11725505 Ki = 1.6 nM T16691 CY1XU6 11729763 Ki = 320 nM T16691 CLYJ75 11729823 Ki = 48.9 nM T16691 C7PVL8 11730467 IC50 = 7780 nM T16691 CMO0I9 11739679 IC50 = 0.8 nM T16691 C2GK7T 11740084 IC50 = 700 nM T16691 C57IKL 11740526 Ki < 1000 nM T16691 CKD26I 11741319 IC50 = 50 nM T16691 CC18PB 11741686 IC50 = 18 nM T16691 C5H0YJ 11743064 IC50 = 126 nM T16691 CPG15O 11743399 IC50 > 1000 nM T16691 CBA17C 11744377 Ki = 10.2 nM T16691 CYV02C 11747350 Ki = 20 nM T16691 C9WO6G 11749539 Ki = 1 nM T16691 CA61BD 11750876 Ki = 57 nM T16691 C3CN0Y 11772625 Ki = 1 nM T16691 CUD91G 11775364 Ki = 8 nM T16691 C0WB7U 11811724 Ki = 490 nM T16691 CAC74F 11820174 Ki = 300 nM T16691 CG3QJ4 11833220 Ki = 260 nM T16691 CZ7Y1I 11849203 Ki = 38 nM T16691 CI4PE1 11849204 Ki = 17 nM T16691 CR8EY5 11849745 Ki = 52 nM T16691 CO0H2M 11849787 Ki = 15 nM T16691 CXLW54 11948707 Ki > 10000 nM T16691 C8JQL7 11957735 IC50 > 10000 nM T16691 C1H2GL 11961315 Ki = 1.7 nM T16691 CSE5A4 11983287 Ki = 1.2 nM T16691 C1QY2P 12005903 Ki = 119 nM T16691 CWE19J 12017572 Ki = 7.4 nM T16691 C2L0RA 12017573 Ki = 9.5 nM T16691 C7RUD8 12017574 Ki = 45 nM T16691 C5TY3Z 12017575 Ki = 93 nM T16691 CV9PF5 12017576 Ki = 183 nM T16691 C9ED3P 12017577 Ki = 5 nM T16691 C5J2UM 12017578 Ki = 154 nM T16691 C6AJ4F 12017579 Ki = 8000 nM T16691 CG56FM 12017580 Ki = 19600 nM T16691 CK28MT 12051078 Ki = 136 nM T16691 CUW18O 12051079 Ki = 300 nM T16691 C8EDN0 12088080 Ki > 1000 nM T16691 C8RB6W 12088082 Ki > 1000 nM T16691 C1QM4J 12147013 Ki = 20 nM T16691 C9RBT8 12147017 Ki = 16 nM T16691 CMH17C 12148615 Ki = 1.8 nM T16691 CEIP49 15480742 Ki = 60 nM T16691 C30CHU 15512229 Ki < 316.23 nM T16691 COWE74 15619875 IC50 = 10 nM T16691 C5QS1J 16019286 IC50 = 1120 nM T16691 CM1EL8 16019288 IC50 = 170 nM T16691 CRM1F0 16019292 Ki = 3.5 nM T16691 C68NQM 16019303 IC50 = 730 nM T16691 CW49DH 16019305 IC50 = 1250 nM T16691 CH03IC 16019310 IC50 = 740 nM T16691 CF0VH8 16019312 IC50 = 220 nM T16691 C1RMU0 16019339 IC50 = 350 nM T16691 CWQ67Z 16019343 IC50 = 820 nM T16691 C0E2AF 16019364 IC50 = 520 nM T16691 CSB0U1 16019366 IC50 = 90 nM T16691 CQTK41 16019372 IC50 = 270 nM T16691 C0PTX8 16019394 IC50 = 960 nM T16691 CTMC92 16019397 IC50 = 650 nM T16691 C8S6VI 16019451 IC50 = 1050 nM T16691 CG5I6Q 16019453 IC50 = 1600 nM T16691 CVW2H6 16019490 IC50 = 1930 nM T16691 C7V4MI 16019508 IC50 = 28.3 nM T16691 CXZ4T7 16019510 IC50 = 1520 nM T16691 CBK40Y 16019514 IC50 = 590 nM T16691 C9IYN1 16019519 IC50 = 710 nM T16691 CD7WK0 16019546 IC50 = 59 nM T16691 CZF0S6 16019548 IC50 = 1170 nM T16691 C4A8GT 16019550 IC50 = 170 nM T16691 C7R0QS 16019553 Ki = 15.9 nM T16691 CHB62Y 16019573 Ki = 28.8 nM T16691 C8GC1T 16019574 IC50 = 690 nM T16691 CL0OT3 16019576 Ki = 1.7 nM T16691 C7T6GI 16019580 Ki = 2.3 nM T16691 C7TP3J 16019601 IC50 = 260 nM T16691 CXMY18 16019602 IC50 = 2010 nM T16691 C3WQ1G 16019604 IC50 = 960 nM T16691 CEP4U1 16019607 IC50 = 1220 nM T16691 CY1JE9 16019609 IC50 = 180 nM T16691 CX2CT6 16019610 IC50 = 140 nM T16691 CL1C5P 16023081 Ki = 88 nM T16691 C3M8GJ 16026344 Ki = 13330 nM T16691 CWY3F2 16037746 Ki = 0.8 nM T16691 CS07QC 16040768 Ki = 32 nM T16691 CX54GY 16049388 Ki = 5.44 nM T16691 CJ1T0W 16070169 Ki = 4.3 nM T16691 CXWC93 16071727 Ki = 6.7 nM T16691 C1SR0O 16071847 Ki = 1.5 nM T16691 CQS4V1 16112801 EC50 = 0.9 nM T16691 CC6Y3J 16116896 Ki = 17 nM T16691 CQ0VT5 16116897 Ki = 28 nM T16691 CA7L8M 16116898 Ki = 9.8 nM T16691 CV6G9J 16116899 Ki = 4.2 nM T16691 C2ATQ4 16116900 Ki = 9.5 nM T16691 CZ1WJ4 16117151 Ki = 1 nM T16691 C4PEY7 16117152 Ki = 2.3 nM T16691 CM32ZX 16117153 Ki = 0.6 nM T16691 CFB1T7 16117154 Ki = 6.7 nM T16691 CJ6D1M 16117278 Ki = 6.3 nM T16691 CXTB90 16117279 Ki = 1 nM T16691 CA23RS 16117280 Ki = 1.5 nM T16691 C8M5KE 16117281 Ki = 3.1 nM T16691 CU9VB2 16117282 Ki = 9.8 nM T16691 C2HI3Q 16117283 Ki = 0.8 nM T16691 C1F2LS 16118795 Ki = 0.7 nM T16691 CT0S9V 16118796 Ki = 3.5 nM T16691 C1BPY5 16118797 Ki = 1.7 nM T16691 C69VDS 16118923 Ki = 1.1 nM T16691 CA0IB2 16118924 Ki = 53 nM T16691 C5DVW2 16118925 Ki = 57 nM T16691 CK4Y1C 16118926 Ki = 44 nM T16691 C76QZH 16118927 Ki = 31 nM T16691 C0PMY8 16118928 Ki = 30 nM T16691 C8OF0W 16118929 Ki = 66 nM T16691 CJ1N3M 16222447 Ki = 15.5 nM T16691 C50ZXQ 16222448 Ki = 8.82 nM T16691 CN16GL 16222450 Ki = 8.28 nM T16691 CGPY68 16222545 Ki = 4.21 nM T16691 C46VQT 16222547 Ki = 1.92 nM T16691 CQ9YZ4 16222548 Ki = 20.4 nM T16691 CK0IB2 16222549 Ki = 1.83 nM T16691 C89XDO 16222651 Ki = 7.5 nM T16691 CSO7W8 16222652 Ki = 5.5 nM T16691 CQC5D4 16222654 Ki = 28.99 nM T16691 CBU75J 16222655 Ki = 16.1 nM T16691 C9HOC0 16222656 Ki = 12.2 nM T16691 C79ADX 16222758 Ki = 18.09 nM T16691 CHOC30 16222759 Ki = 41.1 nM T16691 C5E6MS 16222761 Ki = 15.7 nM T16691 C4HBK5 16222762 Ki = 32.4 nM T16691 CE75KN 16222763 Ki = 15.5 nM T16691 CG8Y3L 16222764 Ki = 43.5 nM T16691 C4XV1Q 16222865 Ki = 32.8 nM T16691 CA2ZJ1 16222866 Ki = 5.89 nM T16691 CQN9G1 16222867 Ki = 19.8 nM T16691 CSJ4H8 16222868 Ki = 15.1 nM T16691 CE0LY9 16222869 Ki = 3.71 nM T16691 C2LDY6 16222870 Ki = 4.57 nM T16691 C1TC5B 16222871 Ki = 13.8 nM T16691 CA6MU9 16222962 Ki = 24.9 nM T16691 CE7QA0 16222963 Ki = 8.13 nM T16691 C9PTN1 16222965 Ki = 7.95 nM T16691 CXZ41D 16223064 Ki = 6.89 nM T16691 CBT9C0 16223065 Ki = 2.68 nM T16691 CN9I4S 16223066 Ki = 24.3 nM T16691 CZ2IS9 16660294 Ki > 10000 nM T16691 C1CER8 16718822 Ki = 17 nM T16691 CD3Q2U 16718826 Ki = 216 nM T16691 C3JV0P 16718827 EC50 = 3.2 nM T16691 C8GOW7 16718869 Ki = 20 nM T16691 C0JQ5W 16718916 Ki = 276 nM T16691 C3YN5S 16718917 EC50 = 0.3 nM T16691 CJ8Y1H 16718919 Ki = 18 nM T16691 CB7G3R 16718920 EC50 = 0.3 nM T16691 C8U4LQ 16718921 Ki = 31 nM T16691 C5MT4H 16718922 Ki = 3 nM T16691 CW03YI 16750338 Ki = 3.8 nM T16691 CT9GP4 16763549 Ki = 2945 nM T16691 C81DEA 16804502 IC50 = 1150 nM T16691 C2F7IH 16956087 IC50 = 540 nM T16691 CZ97JQ 16956089 IC50 = 580 nM T16691 CC8EA5 16956204 IC50 = 930 nM T16691 CR63LE 17055181 Ki = 5100 nM T16691 C0QX5J 17374371 Ki = 11980 nM T16691 CB2J3R 17747575 IC50 > 100 nM T16691 C3BVJ4 17940055 Ki = 31.62 nM T16691 C5D0HA 17940058 Ki = 1.585 nM T16691 CLZ60J 17940080 Ki = 19.95 nM T16691 C1M5VA 17940089 Ki = 1.995 nM T16691 C3UI5Y 17940101 Ki = 0.7943 nM T16691 CBC70F 17940113 Ki = 1.259 nM T16691 CQ96ZT 17940121 Ki = 3.981 nM T16691 C0UE9W 17940125 Ki = 0.3162 nM T16691 C8KJ1Y 17940155 Ki = 1.259 nM T16691 CF46WY 17940169 Ki = 0.5012 nM T16691 CN5G0Y 17940185 Ki = 25.12 nM T16691 CELX94 17940199 Ki = 1.259 nM T16691 C2G6ID 17940212 Ki = 0.631 nM T16691 C6IK5X 17940215 Ki = 0.5012 nM T16691 CG5CO7 17940224 Ki = 1 nM T16691 C92SPR 17940228 Ki = 2.512 nM T16691 CGUS59 17940234 Ki = 7.943 nM T16691 CUS47A 17940243 Ki = 3.162 nM T16691 C6ZM7X 17940245 Ki = 1.995 nM T16691 CL2AS8 17940260 Ki = 1.585 nM T16691 CQC56I 17940268 Ki = 5.012 nM T16691 C9L0AZ 17960999 Ki = 0.3981 nM T16691 CQM7R1 17961002 Ki = 0.631 nM T16691 CR10MN 17961003 Ki = 7.943 nM T16691 CC5SW2 17978373 Ki = 0.3162 nM T16691 C0OL1J 17978376 Ki = 5.012 nM T16691 CH2X5U 17978385 Ki = 25.12 nM T16691 C54VGS 17978406 Ki = 7.943 nM T16691 C3RK0S 17978408 Ki = 0.3162 nM T16691 C6D0PK 18180040 Ki = 2.3 nM T16691 C9PV8A 18180076 IC50 = 13 nM T16691 C6S4JR 18180095 Ki = 1.6 nM T16691 CTA6O3 18180191 Ki = 0.7943 nM T16691 CIZ3C8 18354536 Ki = 0.5012 nM T16691 CXRQ53 18354548 Ki = 0.7943 nM T16691 CHP5L8 18354552 Ki = 3.981 nM T16691 CFT01Z 18354557 Ki = 3.162 nM T16691 C9U3NH 18354572 Ki = 3.981 nM T16691 C2Z9MB 18354574 Ki = 2.512 nM T16691 C37TAU 18354589 Ki = 1.259 nM T16691 CY3P0B 18354590 Ki = 3.981 nM T16691 CV0X4I 18559283 IC50 = 1110 nM T16691 CY0G5A 18559285 IC50 = 890 nM T16691 C0NV6X 18559286 IC50 = 860 nM T16691 C7PKF0 18559353 IC50 = 900 nM T16691 C5LV1E 18559939 IC50 = 5220 nM T16691 CN20SE 18559973 IC50 = 1750 nM T16691 CK74OE 18560047 IC50 > 5000 nM T16691 CC36OB 18560059 IC50 = 1100 nM T16691 CQ4N8G 18560060 IC50 = 1480 nM T16691 CRK34J 18560180 IC50 = 1160 nM T16691 CYWK26 18560181 IC50 = 32 nM T16691 CU93YN 18560182 IC50 = 290 nM T16691 CG56OA 18560184 IC50 = 790 nM T16691 CP24LD 18560186 IC50 = 300 nM T16691 CBH94P 18560202 IC50 = 1380 nM T16691 CW42ZS 18560255 IC50 = 860 nM T16691 COR6X7 18560317 IC50 = 600 nM T16691 C42VJM 18560324 IC50 = 680 nM T16691 CX8HE9 18560325 IC50 = 1330 nM T16691 CE8W5B 18560538 IC50 = 37 nM T16691 C8MWB9 18560539 IC50 = 1370 nM T16691 CP0A5C 18560541 IC50 = 1080 nM T16691 CMPY53 18560542 IC50 = 2030 nM T16691 C7YAO8 18560556 IC50 = 410 nM T16691 C49VTO 18560559 IC50 = 1150 nM T16691 C5SN1R 18560562 IC50 = 280 nM T16691 C6QOH2 18560564 IC50 = 570 nM T16691 C1OL5W 18590273 IC50 = 1190 nM T16691 CRLJ91 18590409 IC50 = 1000 nM T16691 C0J3WX 18590411 IC50 = 1620 nM T16691 C0CAW5 18590413 IC50 = 1950 nM T16691 C2OU9R 18590416 IC50 = 1350 nM T16691 C5VI2L 18590836 IC50 = 3810 nM T16691 CL5BA2 18591074 IC50 = 1430 nM T16691 CD2OR9 18591266 IC50 = 820 nM T16691 C46POT 18591267 IC50 = 780 nM T16691 C3URK4 18591268 IC50 = 29 nM T16691 C9AYF3 18591269 IC50 = 110 nM T16691 C1RCK3 18591271 IC50 = 480 nM T16691 CT01XH 18591272 IC50 = 2500 nM T16691 C7T8JC 19958494 Ki = 7109.5 nM T16691 C6LI5E 19958507 Ki = 4460.7 nM T16691 C0FAH6 20042470 Ki = 9.3 nM T16691 COBR80 20765662 Ki = 1.995 nM T16691 C9ZE0I 20765664 Ki = 0.631 nM T16691 CKNR40 20765669 Ki = 0.5012 nM T16691 CDXS17 20765678 Ki = 12.59 nM T16691 CBY03N 20846175 Ki = 54.95 nM T16691 CEV21N 20901114 IC50 = 1990 nM T16691 CEV8G2 20901115 Ki = 8.1 nM T16691 C25LZY 20901117 Ki = 5.5 nM T16691 CD7TG3 20901118 IC50 = 290 nM T16691 C3KBJ9 20901120 IC50 = 260 nM T16691 C4A1ZK 20901122 IC50 = 600 nM T16691 CK97WL 20901124 IC50 = 820 nM T16691 C13UBY 20901125 IC50 = 500 nM T16691 C1OP7Q 20901126 IC50 = 580 nM T16691 CY9W8X 20901128 IC50 = 250 nM T16691 CNG3I6 20901131 IC50 = 2210 nM T16691 CGZB95 20901132 IC50 = 2030 nM T16691 CH10OK 20901133 IC50 = 590 nM T16691 CGK3J2 20901136 IC50 = 770 nM T16691 CHCW87 20901139 IC50 = 470 nM T16691 CT0C4W 20901141 IC50 = 46 nM T16691 CIT1E8 20901142 IC50 = 750 nM T16691 C2KBV6 20901145 IC50 = 2380 nM T16691 CLF4Y5 20901160 IC50 = 480 nM T16691 CBK05L 20901163 IC50 = 2170 nM T16691 CY3BN2 20901164 IC50 > 5000 nM T16691 C2TRE0 20901169 IC50 = 800 nM T16691 C5MQ0H 20901172 IC50 = 1830 nM T16691 CVG42R 20901177 IC50 > 5000 nM T16691 C2BVW3 20901182 IC50 > 5000 nM T16691 C4MFW3 20901183 IC50 > 5000 nM T16691 CT7FU4 20901186 IC50 = 590 nM T16691 C27ZYB 20901203 IC50 > 5000 nM T16691 CVE0S9 20901207 Ki = 46 nM T16691 C1R9XF 20901210 IC50 = 670 nM T16691 CD3E7L 20901217 IC50 = 170 nM T16691 CGAH45 20901220 IC50 = 1290 nM T16691 CUV3F8 20901229 IC50 = 610 nM T16691 C0OIT1 20901240 IC50 > 5000 nM T16691 CQ4W3Y 20901253 IC50 = 690 nM T16691 CWA26O 20901254 IC50 = 190 nM T16691 CB5D8X 20901255 IC50 = 1040 nM T16691 CLU06V 20901258 IC50 = 1540 nM T16691 C12EZR 20901259 IC50 = 68 nM T16691 CE45NR 20901261 IC50 = 150 nM T16691 CX8EI0 20901263 IC50 = 540 nM T16691 CP0K5O 20901264 IC50 = 60 nM T16691 CEL9U6 20901265 IC50 = 69 nM T16691 CKE98H 20901266 IC50 = 150 nM T16691 C9Z5WA 20901267 IC50 = 2000 nM T16691 CERG41 20901268 IC50 = 150 nM T16691 C5ZRC0 20901270 IC50 = 920 nM T16691 CO0PH4 20901271 IC50 = 1210 nM T16691 C9LWB8 20901273 IC50 = 1070 nM T16691 C5DG2K 20901275 IC50 = 740 nM T16691 CS9Q4E 20901291 IC50 = 1220 nM T16691 C6H9WC 21092408 Ki = 41858718 nM T16691 C0CA1J 21254909 Ki = 16.6 nM T16691 C3T5HF 21509921 Ki = 154.88 nM T16691 CUO9Q1 21512050 IC50 = 40 nM T16691 CG21AX 21514234 Ki = 64 nM T16691 C4B0TN 21557475 Ki = 1966 nM T16691 C36XOS 22028185 Ki = 22 nM T16691 C5JL1M 22028187 Ki = 200 nM T16691 CYS15E 22028199 Ki = 368 nM T16691 CBN84K 22065997 Ki > 10000 nM T16691 C6UXL4 22330705 Ki = 11360 nM T16691 C6G7ZE 22424009 IC50 = 9.6 nM T16691 CZG9S2 22425072 Ki = 6505 nM T16691 CBL97U 22504458 IC50 = 21 nM T16691 CPD8Q7 22549784 Ki = 16550 nM T16691 CAUH46 22557214 Ki = 1.995 nM T16691 C1T4AB 22557219 Ki = 39.81 nM T16691 CAXR08 22557224 Ki = 199.53 nM T16691 CBN2M3 22557235 Ki = 0.0631 nM T16691 C5VA1T 22557241 Ki = 0.1585 nM T16691 CIRF78 22557257 Ki = 10 nM T16691 C03XCL 22557272 Ki = 0.3981 nM T16691 C9W5CD 22557286 Ki = 316.23 nM T16691 CMN2J0 22557287 Ki = 2.512 nM T16691 CH12KP 22557292 Ki = 3.162 nM T16691 C8NR3D 22662986 Ki = 64 nM T16691 CZ7J4B 22857296 Ki = 400 nM T16691 CDL7A8 23288143 Ki = 99 nM T16691 CO1NA8 23624297 Ki = 11.8 nM T16691 CPX21U 23624307 Ki = 0.5 nM T16691 CLI4F8 23624309 Ki = 3.1 nM T16691 CJ2W3A 23625763 Ki = 1 nM T16691 CA5QC2 23625764 Ki = 2.399 nM T16691 CXD3E6 23625925 Ki = 630.96 nM T16691 CJ18ET 23652557 Ki = 10.8 nM T16691 CIY3P0 23652635 Ki = 8.6 nM T16691 CCL15O 23652787 Ki = 9.2 nM T16691 C3YBE2 23652788 Ki = 10.2 nM T16691 CSIP14 23652790 Ki = 10.6 nM T16691 C76LZN 23652861 Ki = 30.1 nM T16691 C4BXD0 23652863 Ki = 82.3 nM T16691 CV74XB 23652922 Ki = 55.3 nM T16691 CKI17V 23652993 Ki = 20.3 nM T16691 CE24HU 23652994 Ki = 30.5 nM T16691 CR6PO0 23653062 Ki = 10.7 nM T16691 CF7VS8 23653130 Ki = 63.5 nM T16691 C6J3NA 23653133 Ki = 15.2 nM T16691 CKW7V5 23653135 Ki = 3.4 nM T16691 CY9TE3 23655287 Ki = 11 nM T16691 C5I8BA 23655288 Ki = 16 nM T16691 CQL1O9 23655289 Ki = 6 nM T16691 C92TKG 23655290 Ki = 21 nM T16691 C5ZH1E 23655462 Ki = 10 nM T16691 C4I2PZ 23655463 Ki = 14 nM T16691 CA29ZB 23655464 Ki = 47 nM T16691 CU6Y4G 23655465 Ki = 1 nM T16691 CEMW69 23655466 Ki = 30 nM T16691 CS1B3A 23655467 Ki = 7 nM T16691 CLD3F4 23655468 Ki = 6 nM T16691 CFRH01 23655469 Ki = 7 nM T16691 CA03MU 23655664 Ki = 31 nM T16691 CNU2X4 23725134 Ki = 1.6 nM T16691 CVLG35 23757269 Ki = 6 nM T16691 CGD1E3 23757270 Ki = 0.8 nM T16691 CN36KF 23786472 Ki = 43 nM T16691 C9KL1S 23815446 Ki = 230 nM T16691 CVE1R9 23815447 Ki = 3 nM T16691 CG6L3F 23844114 Ki = 0.6 nM T16691 C0KM6Q 23872163 Ki = 27 nM T16691 C37QMN 23872164 Ki = 0.6 nM T16691 CC9XE5 23900125 Ki = 34 nM T16691 CQE1N7 23906630 Ki = 5826 nM T16691 CEA76H 23955921 Ki = 90 nM T16691 C7Y6VG 24763349 Ki = 9.6 nM T16691 CT9HL7 24763350 Ki = 55 nM T16691 C4JZ8U 24763351 Ki = 93 nM T16691 CC1N3K 24763352 Ki = 19 nM T16691 CT8BO3 24763353 Ki = 66 nM T16691 CQ64TA 24763354 Ki = 50 nM T16691 CXI4H2 24763355 Ki = 46 nM T16691 CH1UL9 24763429 Ki = 48 nM T16691 CX7CL6 24763430 Ki = 14 nM T16691 CR89US 24768515 Ki = 10.3 nM T16691 CD7CV6 24771120 Ki = 2.3 nM T16691 CGF70N 24771124 Ki = 15 nM T16691 CC6L2F 24771185 Ki = 18 nM T16691 C89WOM 24776044 Ki = 7.92 nM T16691 C0R4EZ 24776942 Ki = 1.8 nM T16691 CV09KG 24777061 Ki = 49 nM T16691 CNWQ34 24777062 Ki = 90 nM T16691 C9E2MV 24777063 Ki = 220 nM T16691 CCEH06 24781896 IC50 > 100 nM T16691 CD86PT 24781897 IC50 > 100 nM T16691 CP7TJ3 24781898 IC50 > 100 nM T16691 CF17PW 24781899 IC50 > 100 nM T16691 C1JSY8 24781900 IC50 > 100 nM T16691 CJI2O1 24782049 IC50 > 100 nM T16691 CK9T1F 24782050 IC50 > 100 nM T16691 C2O7MV 24782051 IC50 > 100 nM T16691 C0G3RV 24782052 IC50 > 100 nM T16691 CR8DV4 24782058 IC50 > 100 nM T16691 CYR67K 24783294 Ki = 7.1 nM T16691 CW20VF 24783295 Ki = 52 nM T16691 C8B7EG 24783296 Ki = 196 nM T16691 C8UQF0 24783550 Ki = 13 nM T16691 CULV50 24783808 Ki = 13 nM T16691 C9LDH4 24783809 Ki = 9.7 nM T16691 C0VKE6 24783810 Ki = 12 nM T16691 CYAU35 24784066 Ki = 41 nM T16691 CN2W9R 24784069 Ki = 54 nM T16691 C38VPE 24784321 Ki = 64 nM T16691 C37OYB 24784323 Ki = 31 nM T16691 CX3KC0 24784325 Ki = 22 nM T16691 CJ73UQ 24784573 Ki = 22 nM T16691 CU40PB 24784575 Ki = 25 nM T16691 CI9T6E 24784577 Ki = 36 nM T16691 C69JES 24784578 Ki = 88 nM T16691 CN52JE 24784824 Ki = 72 nM T16691 C3JSR4 24794436 IC50 = 53 nM T16691 C58AMS 24829343 Ki = 186.5 nM T16691 CDC91N 24839550 Ki = 1737.8 nM T16691 CUW23K 24854106 Ki = 1800 nM T16691 C6BSX7 24855787 Ki = 27.8 nM T16691 C4LC2K 24855826 Ki > 1000 nM T16691 C7ZOP1 24855830 Ki > 1000 nM T16691 CGHZ87 24855831 Ki = 92 nM T16691 C7ZEF0 24856058 Ki = 2.56 nM T16691 CU90ZK 24861250 Ki = 434 nM T16691 C3HK0J 24865725 Ki > 10000 nM T16691 C0O6FX 24865727 Ki = 1584.89 nM T16691 CT7Z5L 24873459 Ki = 0.1995 nM T16691 C6L7KS 24887518 Ki < 3162.28 nM T16691 CI53SE 24893978 Ki = 4100 nM T16691 CJ63YQ 24894055 Ki = 19 nM T16691 CAOF91 24894071 IC50 > 10000 nM T16691 C5EIW1 24965329 Ki = 3.24 nM T16691 CVYJ09 24965330 Ki = 23.41 nM T16691 C5YX0U 24965331 Ki = 8.58 nM T16691 C5S7UA 24965678 Ki = 11.13 nM T16691 C6U2AP 24965679 Ki = 1.43 nM T16691 CY3BJ4 24965680 Ki = 9.89 nM T16691 CFM8C2 24965681 Ki = 29.15 nM T16691 C91FZJ 24966378 Ki = 30.28 nM T16691 CCGJ63 24966381 Ki = 122 nM T16691 CBK7U0 24966733 Ki = 75.3 nM T16691 CG96KI 24966734 Ki = 97.61 nM T16691 C6WD7A 24966736 Ki = 53.62 nM T16691 CJY04G 24966737 Ki = 222 nM T16691 CT47SL 24966738 Ki = 90.71 nM T16691 C1OKR6 24967096 Ki = 27.19 nM T16691 C8HE6A 24967097 Ki = 165 nM T16691 C49BMW 24967099 Ki = 4.82 nM T16691 CJQR84 24967457 Ki = 13.17 nM T16691 CERH27 24968180 Ki = 278 nM T16691 CGX13L 24968181 Ki = 99.7 nM T16691 C8LD4F 24969960 Ki = 10.72 nM T16691 CMC9J2 24970038 Ki = 7.84 nM T16691 C0YK9A 25024144 Ki = 14.6 nM T16691 C02ABD 25024146 Ki = 17.9 nM T16691 C2G8OK 25024148 Ki = 28.2 nM T16691 CEXI24 25024322 Ki = 3.21 nM T16691 CY7AC1 25024326 Ki = 12.4 nM T16691 CJI5U8 25024332 Ki = 11 nM T16691 CO2RU1 25024524 Ki = 5.52 nM T16691 C4YBW2 25024528 Ki = 11.3 nM T16691 CCQ2Y5 25024529 Ki = 8.3 nM T16691 CL83UF 25024530 Ki = 18 nM T16691 CAN16E 25024724 Ki = 3.02 nM T16691 CJX9Q5 25024725 Ki = 3.15 nM T16691 CMD35T 25024726 Ki = 9.33 nM T16691 CP6K8J 25024727 Ki = 2.97 nM T16691 CKEB12 25024729 Ki = 3.36 nM T16691 CQ3ZF4 25024731 Ki = 4.16 nM T16691 CRYA79 25024924 Ki = 2.58 nM T16691 CCF9K4 25024926 Ki = 7.77 nM T16691 C90GZM 25024928 Ki = 5.57 nM T16691 CW6QY9 25024930 Ki = 2.52 nM T16691 CSCP07 25025118 Ki = 14.9 nM T16691 CQ3P5R 25025314 Ki = 5.81 nM T16691 C1PKF0 25056080 Ki = 24.1 nM T16691 CYJ5G1 25067564 Ki = 4.46 nM T16691 CBY3O2 25070582 IC50 = 1800 nM T16691 C4GSD8 25110702 Ki = 1.585 nM T16691 CR17NY 25110703 Ki = 2.512 nM T16691 CNS84K 25117676 Ki = 0.51 nM T16691 C4WV0K 25117677 IC50 = 17.5 nM T16691 CL19XF 25117679 Ki = 21.1 nM T16691 CWFY19 25117680 Ki = 13.7 nM T16691 CSW9K6 25117681 Ki = 36.9 nM T16691 C1PG8Z 25122651 Ki = 4.27 nM T16691 CD3R5U 25122652 Ki = 3.62 nM T16691 CK58IM 25122653 Ki = 4.52 nM T16691 CA12QG 25122654 Ki = 8.04 nM T16691 C3M0EY 25123011 Ki = 18.22 nM T16691 CZX2R0 25123012 Ki = 13.09 nM T16691 CNV98C 25123013 Ki = 3.55 nM T16691 C3N6SM 25123014 Ki = 3.06 nM T16691 CDQ70A 25208878 EC50 = 14 nM T16691 CJ1Z9H 25216680 Ki > 10000 nM T16691 C1T3LR 25218143 Ki > 10000 nM T16691 CPI03N 25218397 Ki > 10000 nM T16691 CL1R3Q 25218401 Ki > 10000 nM T16691 CLIZ27 25251903 Ki = 8883 nM T16691 CM2T9Y 25263297 Ki = 7.9 nM T16691 CR5D2U 25263298 Ki = 50 nM T16691 CR5JL8 25263299 Ki = 1.2 nM T16691 C9G3TC 25263300 Ki = 1.8 nM T16691 CAF19L 25263301 Ki = 2.1 nM T16691 CFJM71 25263302 Ki = 1.3 nM T16691 C5IB8J 25263304 Ki = 10.3 nM T16691 CUBL21 25263305 Ki = 0.6 nM T16691 C8BV1Y 25263306 Ki = 15.3 nM T16691 CM2P4B 25263307 Ki = 11.6 nM T16691 CP25TS 25263308 Ki = 9.3 nM T16691 CUT3O9 25263309 Ki = 61.6 nM T16691 CK0UJ9 25263310 Ki = 126 nM T16691 CAH0F1 25263311 Ki = 45.6 nM T16691 C73QEX 25263312 Ki = 70.7 nM T16691 C18HPB 25263313 Ki = 2.5 nM T16691 C0RK3L 25263314 Ki = 3.3 nM T16691 CFK36A 25263315 Ki = 174 nM T16691 C18PIH 25263316 Ki = 92.5 nM T16691 C1DS3N 25263317 Ki = 42 nM T16691 C0W3ZY 25263318 Ki = 219 nM T16691 CZ69DU 25263319 Ki > 440 nM T16691 C15QMB 25263320 Ki = 6.9 nM T16691 CQH59C 25263321 Ki = 39.8 nM T16691 C1XZ9U 25263322 Ki = 2.8 nM T16691 C1GPQ9 25263323 Ki = 39.5 nM T16691 CP50YT 25263324 Ki = 17.9 nM T16691 C2HJ4M 25263325 Ki > 440 nM T16691 CJQ87U 25263326 Ki = 8.1 nM T16691 C8QS7R 25263327 Ki = 17.8 nM T16691 CPK94B 25263328 Ki = 19.1 nM T16691 CI4OU7 25263329 Ki > 440 nM T16691 CC89NU 25263330 Ki = 50 nM T16691 C56YFT 25263331 Ki > 440 nM T16691 CK7JV5 25263332 Ki > 440 nM T16691 C5XZ3Y 25263333 Ki = 239 nM T16691 CPV78N 25263334 Ki = 48.5 nM T16691 CFCT24 25263335 Ki > 440 nM T16691 C06CZE 25263336 Ki = 10.5 nM T16691 C52XBP 25263337 Ki = 208 nM T16691 CD9HU0 25263338 Ki = 6.4 nM T16691 CTUR83 25263339 Ki = 2.4 nM T16691 CJ69LP 25263340 Ki = 4.3 nM T16691 C5FQW4 25263341 Ki > 440 nM T16691 C0LNU7 25263342 Ki = 3.5 nM T16691 C5A1YV 25263343 Ki = 6.5 nM T16691 C8CMO5 25263344 Ki = 19.6 nM T16691 CQP58M 25263345 Ki = 26.1 nM T16691 CN4JF1 25263346 Ki = 18.4 nM T16691 C3OIN1 25263347 Ki = 5.8 nM T16691 CJ2LH8 25263348 Ki = 24.7 nM T16691 C3RQW5 25263349 Ki = 13.6 nM T16691 CX63AQ 25263350 Ki = 10.1 nM T16691 CPE2C1 25263351 Ki = 15.1 nM T16691 CLNE06 25263352 Ki = 28.9 nM T16691 CUE1X8 25263353 Ki = 11.3 nM T16691 C15JZS 25263354 Ki = 1.5 nM T16691 CFDT07 25263355 Ki = 2.7 nM T16691 CG56DF 42388639 IC50 = 2634 nM T16691 CH5QX6 42389467 IC50 > 10000 nM T16691 COBT83 42602875 Ki < 10 nM T16691 CY7W2J 42631003 Ki = 1.2 nM T16691 CV2X5B 42635027 IC50 = 2839 nM T16691 CS9Q3H 42635204 IC50 = 1956 nM T16691 CQ2M5S 42635387 IC50 = 768 nM T16691 CR3KM7 42635388 IC50 = 6925 nM T16691 CJ3NP5 42636941 IC50 > 10000 nM T16691 CJ41QV 44126269 Ki = 2.399 nM T16691 CG1VP5 44126270 IC50 = 1050 nM T16691 CN3IA4 44126272 IC50 = 974 nM T16691 CY6PC2 44126325 IC50 = 666 nM T16691 C32MRX 44126326 IC50 = 977 nM T16691 CQ28AG 44126327 IC50 = 4070 nM T16691 CNF19Z 44126328 IC50 = 2270 nM T16691 CHFE79 44126329 IC50 = 860 nM T16691 C2Q0UX 44126330 IC50 = 440 nM T16691 CV4TD7 44155107 Ki = 0.549 nM T16691 C6TND7 44155109 Ki = 0.44 nM T16691 CEZ18Q 44155871 Ki = 22.2 nM T16691 C1VF8H 44155874 Ki = 1.2 nM T16691 C1LJY7 44155875 Ki = 1.91 nM T16691 C2Z6PY 44155876 Ki = 6.761 nM T16691 CEJY41 44155992 Ki = 1.072 nM T16691 CE41VX 44155994 Ki = 0.7586 nM T16691 CA5N1Z 44156502 Ki = 14.5 nM T16691 CH68EA 44156622 Ki = 0.3981 nM T16691 C91MAJ 44156624 Ki = 0.5012 nM T16691 C97EQS 44156626 Ki = 0.1862 nM T16691 CXM4K7 44156628 Ki = 0.088 nM T16691 CY41DQ 44156752 Ki = 0.202 nM T16691 C73FZD 44156754 Ki = 0.112 nM T16691 CNXV95 44156756 Ki = 0.49 nM T16691 CPE0L5 44156863 Ki = 0.458 nM T16691 C2SYR0 44216882 Ki = 1.5 nM T16691 CPI9X4 44224259 IC50 = 5990 nM T16691 CR0W9C 44240753 Ki = 7.1 nM T16691 CC4A6H 44240802 Ki = 25 nM T16691 CN1UZ6 44240860 Ki = 11.6 nM T16691 CA8GC6 44242965 Ki = 48 nM T16691 CA9E6X 44248103 Ki = 3.83 nM T16691 C2FDB1 44250364 IC50 > 10000 nM T16691 C8MC0Q 44251387 IC50 > 10000 nM T16691 C5YEA8 44251388 IC50 > 10000 nM T16691 C0BSF6 44251389 IC50 > 10000 nM T16691 CL09IQ 44263496 Ki = 80 nM T16691 C87MXH 44263497 Ki = 64 nM T16691 CB0OX8 44263956 Ki = 510 nM T16691 CC2OD4 44278111 Ki > 10000 nM T16691 CRMA84 44278114 Ki = 6486.5 nM T16691 CF0Y4M 44278115 Ki > 10000 nM T16691 CMI97L 44292800 Ki = 4.7 nM T16691 CKQ5B7 44293023 Ki = 3.3 nM T16691 CL8GV9 44293077 Ki = 3.6 nM T16691 C7PC8W 44327453 Ki = 130 nM T16691 C6MU4R 44327527 Ki = 7.2 nM T16691 CG06CL 44327759 Ki = 0.3 nM T16691 CER86D 44327952 Ki = 180 nM T16691 CQC8S9 44327972 Ki = 33 nM T16691 C5QXL8 44327999 Ki = 6.9 nM T16691 C59TSH 44328120 Ki = 50.12 nM T16691 C6BMZ7 44328589 Ki = 79.43 nM T16691 CU89ZL 44328649 Ki = 31.62 nM T16691 CU2Z3F 44328732 Ki = 1.995 nM T16691 CNHP91 44328748 Ki = 5.012 nM T16691 C02WXU 44341344 Ki = 23 nM T16691 CUXH48 44352308 Ki = 1770 nM T16691 C3LKN1 44364048 Ki = 125.89 nM T16691 CQ07ZJ 44369364 Ki = 3.981 nM T16691 C52GZW 44369415 Ki = 0.7943 nM T16691 C4B3EU 44369594 Ki = 1.995 nM T16691 C5MF9A 44369599 Ki = 158.49 nM T16691 CPQ84Z 44369828 Ki = 3.162 nM T16691 C3LD8S 44369855 Ki = 2.512 nM T16691 CV1O8R 44369858 Ki = 2.512 nM T16691 C3YSZ1 44386408 Ki = 9.4 nM T16691 CZOG07 44386469 Ki = 47 nM T16691 CZQK94 44386665 Ki = 6000 nM T16691 CX05UV 44386717 Ki = 2 nM T16691 C6WJ7D 44386718 Ki = 14 nM T16691 C4IFL1 44386772 Ki = 29 nM T16691 CTP90D 44386815 Ki = 6000 nM T16691 CB72DR 44386821 Ki = 5.1 nM T16691 C83PMF 44386822 Ki = 7.6 nM T16691 C57ANV 44386851 Ki = 200 nM T16691 C9NS0P 44386911 Ki = 5 nM T16691 C48ZFS 44387089 Ki = 2.4 nM T16691 C7VJO9 44387804 Ki = 57.7 nM T16691 CQCJ32 44387817 Ki = 117 nM T16691 CXD1R3 44388701 Ki = 1.4 nM T16691 CX8GB0 44388943 Ki = 1 nM T16691 CCA46R 44388944 Ki = 7 nM T16691 C4FBC2 44388950 Ki = 3 nM T16691 CPW47O 44388951 Ki = 3 nM T16691 C2AS1M 44388953 Ki = 31 nM T16691 CCX5P2 44388954 Ki = 118 nM T16691 CT50YA 44388955 Ki = 20 nM T16691 CTPG47 44388956 Ki = 3 nM T16691 CVE02M 44388970 Ki = 5 nM T16691 CNAH73 44388971 Ki = 246 nM T16691 CJVF20 44388980 Ki = 50 nM T16691 C7UO3A 44388986 Ki = 54 nM T16691 C1XJR3 44388987 Ki = 29 nM T16691 C6FWJ7 44388999 Ki = 2 nM T16691 CKWI18 44389001 IC50 = 0.7 nM T16691 C6QG9Z 44389002 IC50 = 3.9 nM T16691 CQ85AW 44389003 Ki = 0.4 nM T16691 C3LRC0 44389004 Ki = 1 nM T16691 CCV4R6 44389010 Ki = 27 nM T16691 CW25QI 44389015 Ki = 1 nM T16691 C8AG7U 44389016 Ki = 1 nM T16691 C5Q2DG 44389023 IC50 = 4.1 nM T16691 C0C6AK 44389024 Ki = 77 nM T16691 CW2VL5 44389025 Ki = 2.4 nM T16691 C3TQF5 44389074 Ki = 3 nM T16691 C0Y1WT 44389075 Ki = 14 nM T16691 C9Q8HJ 44389081 IC50 = 1.3 nM T16691 CMK43D 44389086 Ki = 20 nM T16691 C6F0PN 44389091 Ki = 18 nM T16691 CI29MW 44389099 Ki = 4 nM T16691 C49POD 44389999 Ki = 63 nM T16691 CEP37C 44390011 Ki = 57 nM T16691 C8EO5M 44390023 Ki = 35 nM T16691 CCS1R5 44390045 Ki = 21 nM T16691 CD27FB 44390095 Ki = 54 nM T16691 CRE63B 44390105 Ki = 190 nM T16691 CG9S1O 44393045 Ki = 172 nM T16691 CO6EY0 44393113 Ki = 380 nM T16691 CFZ06U 44395451 Ki = 5.7 nM T16691 C2YT8F 44395458 Ki = 1011 nM T16691 CWP5C1 44395499 Ki = 27 nM T16691 CDWH09 44395500 Ki = 15.5 nM T16691 CWV3T0 44395570 Ki = 23 nM T16691 C28QOZ 44395595 Ki = 5 nM T16691 CIVS89 44395604 Ki = 57 nM T16691 CK9QF8 44395632 Ki = 46 nM T16691 CG1P9D 44395633 Ki = 42 nM T16691 CGH8T3 44395663 Ki = 44 nM T16691 CM4Q5J 44395664 IC50 = 23 nM T16691 CL70AX 44396965 Ki = 2400 nM T16691 C2CV9R 44397117 Ki = 550 nM T16691 CWH17E 44397119 Ki = 29 nM T16691 C2H4SK 44397258 Ki = 8750 nM T16691 CA2M3N 44397322 Ki = 9.9 nM T16691 C21NVO 44397392 Ki = 7.8 nM T16691 CW3D4Z 44397420 Ki = 640 nM T16691 CA0G3Y 44397550 Ki = 27.7 nM T16691 C4B0OI 44397588 Ki < 7943.28 nM T16691 C5FP0R 44397589 Ki < 1995.26 nM T16691 CD6JC7 44397650 Ki = 9.1 nM T16691 CE3G8U 44397670 Ki = 3981.07 nM T16691 C51HTB 44397689 Ki = 1.7 nM T16691 C5FG9Z 44398251 Ki = 5.012 nM T16691 CGXA61 44398325 Ki = 0.7943 nM T16691 CZT23U 44398389 Ki = 0.1995 nM T16691 CMW7N1 44398420 Ki = 79.43 nM T16691 C7FJ9V 44398455 Ki = 63.1 nM T16691 CZ86NU 44398555 Ki = 39.81 nM T16691 CSA67D 44398568 Ki = 3.162 nM T16691 CXH9F6 44398569 Ki = 251.19 nM T16691 C25PRL 44398570 Ki = 1 nM T16691 C2J7IK 44398571 Ki = 0.1259 nM T16691 CK19DL 44398577 Ki = 6.31 nM T16691 CKB7D0 44401278 Ki = 100 nM T16691 CZOP35 44401434 Ki = 57 nM T16691 C9XM1K 44401465 Ki = 50 nM T16691 C4UG8Z 44403044 IC50 = 1 nM T16691 CE10DO 44403046 Ki = 9.8 nM T16691 C6D7PC 44403047 Ki = 3 nM T16691 CV4I3H 44403048 Ki = 11 nM T16691 C53GTV 44403052 Ki = 43 nM T16691 CU42TN 44403053 Ki = 22 nM T16691 C3G0NR 44403055 Ki = 4.6 nM T16691 COC2X7 44403056 Ki = 49 nM T16691 C42TYP 44403057 Ki = 34 nM T16691 CD71OL 44403059 Ki = 9.2 nM T16691 C5NS1R 44403060 Ki = 13 nM T16691 CS6QR7 44403061 Ki = 33 nM T16691 C2VJK8 44403062 Ki = 40 nM T16691 C4SI2K 44403063 Ki = 21.7 nM T16691 C7GNI8 44403064 Ki = 8.5 nM T16691 CNV08U 44403065 Ki = 7 nM T16691 C0MDT3 44403066 Ki = 49 nM T16691 CAE0Q4 44403070 Ki = 14 nM T16691 C8FH9R 44403071 Ki = 44.7 nM T16691 CCKI37 44403072 Ki = 10.5 nM T16691 CA5HK9 44403073 Ki = 23 nM T16691 CM04HK 44403074 Ki = 25 nM T16691 C6JG7H 44403075 Ki = 22 nM T16691 C5CHG2 44403076 Ki = 16 nM T16691 C1FJK7 44403077 Ki = 20 nM T16691 CHJ21O 44403078 Ki = 283.7 nM T16691 CRGK10 44403079 Ki = 252.7 nM T16691 CT0K6J 44403080 Ki = 41.7 nM T16691 CK5B2Y 44403082 Ki = 13 nM T16691 C69KGB 44403083 Ki = 20 nM T16691 CJ3NF1 44403084 Ki = 4 nM T16691 CUF3Y7 44403085 Ki = 271.3 nM T16691 CYPN60 44403086 Ki = 116 nM T16691 CN76UV 44403087 Ki = 26 nM T16691 CB9N2C 44403088 Ki = 48 nM T16691 C2U5VA 44403089 Ki = 7 nM T16691 C1D5XJ 44403090 Ki = 22.7 nM T16691 C7DI0U 44403091 Ki = 58 nM T16691 CT5J9L 44403092 Ki = 4 nM T16691 CM52PQ 44403093 Ki = 7 nM T16691 C0MJ5E 44403094 Ki = 1.5 nM T16691 C1B4QL 44403095 Ki = 5089 nM T16691 C78XLE 44403096 Ki = 8 nM T16691 C8JVC0 44403097 Ki = 3 nM T16691 C1YL7Z 44403098 Ki > 10000 nM T16691 C2F3PA 44403099 Ki = 5 nM T16691 CJE43P 44403100 Ki = 19.3 nM T16691 CFV98A 44403101 Ki = 1429 nM T16691 C6OY9S 44403102 Ki = 2863 nM T16691 CZYP63 44403103 Ki = 3 nM T16691 CUS27C 44403104 IC50 = 7.3 nM T16691 CH4SX6 44403105 Ki > 10000 nM T16691 CK73IG 44403277 Ki = 7.943 nM T16691 CK8ZC2 44403297 Ki = 1 nM T16691 CU20KD 44403304 Ki = 0.631 nM T16691 CGV60Z 44403305 Ki = 0.3981 nM T16691 CCR38V 44403327 Ki = 0.5012 nM T16691 C93VWG 44403335 IC50 = 90 nM T16691 CDR8Y4 44403351 IC50 = 40 nM T16691 CC4X2L 44403358 IC50 = 30 nM T16691 CNE30I 44403366 IC50 = 40 nM T16691 CQ98FN 44403367 IC50 = 100 nM T16691 CMUH71 44403375 IC50 = 30 nM T16691 CQH74S 44403376 IC50 = 60 nM T16691 CGMD49 44403377 IC50 = 50 nM T16691 C6WB0T 44403384 IC50 = 70 nM T16691 CBX76M 44403386 IC50 = 600 nM T16691 C4LKC1 44404394 Ki = 469 nM T16691 C3EJ4G 44404396 Ki = 841 nM T16691 C6NEJ8 44405348 Ki = 7 nM T16691 C9T0GF 44405357 Ki = 1.9 nM T16691 CJB4D6 44405369 Ki = 26 nM T16691 CE5N7Y 44405385 Ki = 21 nM T16691 CG87PW 44409290 Ki > 720 nM T16691 CI3F8D 44413493 Ki = 210 nM T16691 COC47A 44413644 Ki = 165 nM T16691 CS01VM 44413645 Ki = 205 nM T16691 C8XO7Q 44420490 Ki = 14 nM T16691 CB7L2P 44420491 Ki = 11 nM T16691 CJIP85 44420568 Ki = 106 nM T16691 C0TC1M 44420569 Ki = 15 nM T16691 CE2V0S 44425698 Ki = 50.12 nM T16691 C2TE3S 44425699 Ki = 5.012 nM T16691 CU52GB 44425701 Ki = 1.259 nM T16691 C9F1XP 44425702 Ki = 7.943 nM T16691 CR1QN5 44425703 Ki = 25.12 nM T16691 C5UZS7 44425704 Ki = 6.31 nM T16691 CN96FA 44425705 Ki = 10 nM T16691 C1J9MY 44425706 Ki = 15.85 nM T16691 CPI52U 44425708 Ki = 12.59 nM T16691 CNZ3M7 44425711 Ki = 50.12 nM T16691 C92AZG 44425714 Ki = 50.12 nM T16691 C7LP1B 44425717 Ki = 31.62 nM T16691 CX8TR0 44425719 Ki = 7.943 nM T16691 CZ3RM2 44435219 Ki = 9900 nM T16691 C6NA0Z 44435538 IC50 = 9.6 nM T16691 CFZ43E 44435603 Ki = 1.995 nM T16691 C2NUK7 44435604 Ki = 2.692 nM T16691 C64YGX 44435607 Ki = 8.5 nM T16691 CU8MX9 44435608 Ki = 1.5 nM T16691 CEL2F1 44435609 Ki = 5.495 nM T16691 CGJX16 44435610 Ki = 1.288 nM T16691 CB0A9Z 44435612 Ki = 4.266 nM T16691 C0HBD2 44435613 Ki = 1.288 nM T16691 C4SC3H 44435614 Ki = 2.5 nM T16691 C7K9LY 44435615 Ki = 5.6 nM T16691 CR2U0J 44435616 Ki = 1.4 nM T16691 CO6YJ3 44435617 Ki = 5 nM T16691 CCK8S6 44435618 Ki = 2.188 nM T16691 CI07QG 44435619 Ki = 1.5 nM T16691 CO9S3E 44435620 Ki = 4.169 nM T16691 C5K3CJ 44435621 Ki = 0.8913 nM T16691 CN9T5I 44435622 Ki = 10.96 nM T16691 C5WQ7O 44435623 Ki = 8.3 nM T16691 CYCH81 44435624 Ki = 3.3 nM T16691 COS74A 44435625 Ki = 1 nM T16691 CB2O6F 44435626 Ki = 5.7 nM T16691 CIB4M5 44435627 Ki = 4.898 nM T16691 C8UW3X 44435628 Ki = 3.7 nM T16691 CW9SM4 44435629 Ki = 1.288 nM T16691 C2L6RY 44435630 Ki = 7.586 nM T16691 CL02YH 44435631 Ki = 11.48 nM T16691 CL2M7U 44435632 Ki = 33.11 nM T16691 CA09IP 44435633 Ki = 11.1 nM T16691 CD4M9E 44435635 Ki = 4.571 nM T16691 CEA1M2 44435637 Ki = 12 nM T16691 C8S1WD 44435638 Ki = 2.089 nM T16691 C1WX0B 44435639 Ki = 3.8 nM T16691 CSQ21Z 44435640 Ki = 1.995 nM T16691 C9JR1U 44435641 Ki = 4.677 nM T16691 CD8GO7 44435642 Ki = 4.365 nM T16691 CY27QR 44435643 Ki = 3.388 nM T16691 C8H5MA 44435644 Ki = 9.333 nM T16691 C8GY6Q 44435646 Ki = 6.1 nM T16691 CSHJ16 44435647 Ki = 3.89 nM T16691 C9P1AJ 44435649 Ki = 13.49 nM T16691 CL13NV 44435650 Ki = 1.2 nM T16691 CC1I9Y 44435652 Ki = 1.9 nM T16691 CC5G9M 44435653 Ki = 3.2 nM T16691 CS6HP4 44438689 Ki = 590 nM T16691 C6D5OV 44438708 Ki = 280 nM T16691 C3HJY2 44438709 Ki = 135 nM T16691 C0V6QX 44438711 Ki = 220 nM T16691 C54RZL 44438716 Ki = 440 nM T16691 CH0YR3 44438718 Ki = 210 nM T16691 CJ9IW7 44438720 Ki = 13 nM T16691 CI9BD3 44438722 Ki = 1.9 nM T16691 C7R1IF 44438723 Ki = 94 nM T16691 CY9B7P 44438726 Ki = 29 nM T16691 C4UCP2 44438728 Ki = 132 nM T16691 C2I9YU 44438729 Ki = 44 nM T16691 C6R3CH 44438731 Ki = 445 nM T16691 CYZ2F7 44438732 Ki = 20 nM T16691 C0YE5U 44438738 Ki = 1.5 nM T16691 C4U5VN 44438743 Ki = 6000 nM T16691 CKZF16 44439165 Ki = 7943.28 nM T16691 CA4HZ3 44439167 Ki < 10000 nM T16691 C6R7JW 44441237 Ki = 1.259 nM T16691 CE95NG 44441238 Ki = 630.96 nM T16691 CD7WK4 44441239 Ki = 3.981 nM T16691 CP3V1M 44441240 Ki = 3.981 nM T16691 C8E3UZ 44441241 Ki = 5.012 nM T16691 CMY15F 44441242 Ki = 125.89 nM T16691 C3F8TA 44443506 Ki = 402 nM T16691 CNBC07 44443511 Ki = 1888 nM T16691 CO6R9T 44446213 Ki = 293 nM T16691 C6PR5Y 44446214 Ki = 893 nM T16691 CZL97F 44455426 Ki = 3890 nM T16691 C6BFI0 44456033 Ki = 1028.4 nM T16691 C12XGE 44456400 Ki > 10000 nM T16691 CS79YN 44459048 Ki = 42.66 nM T16691 C4DL5C 44469677 IC50 > 10000 nM T16691 CM5EY8 44474470 Ki = 26 nM T16691 C8UON6 44474625 Ki = 5.2 nM T16691 C6HVU1 44474629 Ki = 1.2 nM T16691 CE2Z8S 44474631 Ki = 2.6 nM T16691 C8LA4W 44474797 Ki = 4.1 nM T16691 CMST50 44476434 Ki = 1.9 nM T16691 CXY7T9 44476436 Ki = 0.39 nM T16691 CPX32Z 44476514 Ki = 0.68 nM T16691 C6V2YR 44476607 Ki = 0.82 nM T16691 C3F8HQ 44476611 Ki = 2.1 nM T16691 C2WXT0 44476704 Ki = 60.4 nM T16691 C8QCU7 44476801 Ki = 372 nM T16691 CO5SX2 44476804 Ki = 1155 nM T16691 C1H8NX 44516817 Ki = 0.2 nM T16691 C3D4HR 44537940 Ki = 7.5 nM T16691 CJ7U3K 44554227 Ki = 2.9 nM T16691 CT67VS 44554228 Ki = 2.2 nM T16691 CM0I1P 44554393 Ki = 4.6 nM T16691 CXDZ28 44554394 Ki = 1.9 nM T16691 CNHA47 44554395 Ki = 1.6 nM T16691 CA5G3B 44567932 Ki = 193 nM T16691 C3PZE4 44567933 Ki = 33 nM T16691 CJBD54 44567981 Ki = 23 nM T16691 CRM8G3 44567982 Ki = 19 nM T16691 COB09W 44567983 Ki = 41 nM T16691 CS5X2K 44567984 Ki = 18 nM T16691 C65HIW 44567985 Ki = 68 nM T16691 CRG8E2 44568019 Ki = 89 nM T16691 CGU0L3 44568020 Ki = 46 nM T16691 CFKG06 44568021 Ki = 24 nM T16691 CU3SX6 44568022 Ki = 33 nM T16691 C8WC9P 44568061 Ki = 12 nM T16691 CV0RZ9 44568062 Ki = 19 nM T16691 CGD81I 44568063 Ki = 50 nM T16691 CPYC85 44568064 Ki = 124 nM T16691 C7LZ4X 44568065 Ki = 85 nM T16691 C20LPH 44568101 Ki = 139 nM T16691 C3RFT5 44568102 Ki = 504 nM T16691 C3UX9P 44568103 Ki = 324 nM T16691 C8M0YW 44568104 Ki = 253 nM T16691 CN8M2K 44568139 Ki = 12 nM T16691 C68JSG 44579085 Ki = 1.585 nM T16691 CVU2Z0 44579129 Ki = 7.943 nM T16691 C4PJ7T 44579130 Ki = 7.943 nM T16691 CEH1N0 44579131 Ki = 1.995 nM T16691 CW69AF 44579132 Ki = 100 nM T16691 CM1PH0 44579133 Ki = 7.943 nM T16691 CL3J1S 44579180 Ki = 3.981 nM T16691 C4N2PZ 44579181 Ki = 1.259 nM T16691 C74XJR 44579182 Ki = 1.995 nM T16691 C9PY2D 44579183 Ki = 39.81 nM T16691 C5NS6H 44581972 Ki = 489.78 nM T16691 CK8Z1P 44581973 Ki = 831.76 nM T16691 C3UQ9Z 44581974 Ki = 3388.44 nM T16691 CRCH48 44582675 Ki = 3842 nM T16691 CEJ4R8 44582676 Ki > 10000 nM T16691 CZGP86 44582677 Ki > 10000 nM T16691 C5QB4K 44582678 Ki > 10000 nM T16691 C01RCI 44582705 Ki > 10000 nM T16691 CXL25V 44582706 Ki > 10000 nM T16691 C8MR1X 44582707 Ki > 10000 nM T16691 C4IT1N 44582708 Ki > 10000 nM T16691 C18APH 44591028 Ki = 176 nM T16691 C8C2RL 44591029 Ki = 127 nM T16691 C0TGD4 44591068 Ki = 33 nM T16691 CQU75A 44591069 Ki = 79 nM T16691 C6RYT5 44591592 Ki = 4 nM T16691 C5JN4B 44591611 Ki = 3.2 nM T16691 CB0S4Z 44592109 IC50 > 10000 nM T16691 CQI0D4 45102707 Ki = 158.49 nM T16691 CSEP-69 45102708 Ki = 630.96 nM T16691 C0DLU3 45109862 IC50 = 1412 nM T16691 C1AM5U 45113275 IC50 = 26000 nM T16691 CH0BX2 45113399 IC50 = 62000 nM T16691 CGB2Z0 45113400 Ki = 2.1 nM T16691 C50CMH 45113401 IC50 = 3900 nM T16691 CWE53Z 45113403 IC50 = 85 nM T16691 CHN63A 45113404 IC50 = 3400 nM T16691 CCVA63 45113530 Ki = 5.7 nM T16691 CR52JD 45113534 IC50 = 620 nM T16691 C7I2OM 45113535 IC50 = 28000 nM T16691 CZ71RN 45278805 IC50 = 713 nM T16691 CZN6M7 45278882 IC50 = 1904 nM T16691 CPEY83 45378934 Ki = 54.3 nM T16691 CU36SC 45378935 Ki = 48.7 nM T16691 CHNI56 45378936 Ki = 75.8 nM T16691 C0CHF4 45482789 IC50 = 9580 nM T16691 CD5H2X 45483622 Ki = 2.2 nM T16691 C1BQT4 45483628 Ki = 70 nM T16691 C4IY7C 45483630 Ki <= 8 nM T16691 C5O1SN 45483634 Ki <= 8 nM T16691 CNLO32 45484297 Ki = 4.7 nM T16691 C28VBH 45484298 Ki = 11.7 nM T16691 C0VI9E 45484299 Ki = 9 nM T16691 C0C2LY 45484307 Ki = 15 nM T16691 CK1CD7 45484322 Ki = 3.3 nM T16691 CHI36F 45484332 Ki = 88 nM T16691 C3JZC6 45484333 Ki = 0.9 nM T16691 CAM93H 45484339 Ki = 45 nM T16691 CCB6J0 45484340 Ki = 0.9 nM T16691 C6YO5M 45484352 EC50 = 30 nM T16691 C0Z8VW 45484381 Ki = 4.2 nM T16691 C1IBR5 45484382 Ki = 4.7 nM T16691 CU0YM2 45484383 Ki = 2.1 nM T16691 C83ZJN 45484384 Ki = 2.1 nM T16691 CGZW45 45484398 Ki = 4.3 nM T16691 CYS1T3 45484399 Ki = 2.9 nM T16691 CKYS61 45487099 Ki = 46 nM T16691 C4M9EL 45487100 Ki = 42 nM T16691 CZ4E6T 45487112 Ki = 214 nM T16691 CI7S4B 45487113 Ki = 56 nM T16691 C8PGH3 45487128 Ki = 11.3 nM T16691 CBF24J 45487129 Ki = 3.9 nM T16691 CO81XT 45487139 Ki = 1.7 nM T16691 C7HN5G 45487140 Ki = 76 nM T16691 CL2JK1 45487150 Ki = 35 nM T16691 CH90CZ 45488126 Ki > 1000 nM T16691 CG9U2R 45488130 Ki > 1000 nM T16691 C7N4GP 45488138 Ki > 1000 nM T16691 CH29KP 45488139 Ki = 16 nM T16691 CDAJ27 45488143 Ki = 16 nM T16691 CZYC01 45488151 Ki = 13 nM T16691 C8PH0Y 45488152 Ki = 5 nM T16691 CC2OU0 45488156 Ki > 1000 nM T16691 CL4G8T 45488165 Ki = 27 nM T16691 C5NDO6 45488166 Ki = 17 nM T16691 C0GMN4 45488171 Ki > 1000 nM T16691 C3ZAL4 45488172 Ki > 1000 nM T16691 C3PYL9 45488174 Ki > 1000 nM T16691 CFT7C5 45488175 Ki > 1000 nM T16691 CX1A2N 45488179 Ki > 1000 nM T16691 CA8I7U 45488180 Ki > 1000 nM T16691 C01QBM 45488181 Ki > 1000 nM T16691 COX47A 45488183 Ki > 1000 nM T16691 C8ETO2 45488184 Ki > 1000 nM T16691 C5KOL1 46189932 Ki = 0.5248 nM T16691 CQ8I3H 46189935 Ki = 0.6457 nM T16691 CD2Y4X 46189980 Ki = 1.38 nM T16691 C1YO4C 46189984 Ki = 0.5495 nM T16691 CI30OJ 46189987 Ki = 1.413 nM T16691 CF3WR6 46190034 Ki = 0.7079 nM T16691 C71HDV 46190037 Ki = 0.4169 nM T16691 C2DF3H 46190041 Ki = 2.089 nM T16691 C5KRC3 46203710 Ki = 0.53 nM T16691 CIV92F 46214153 Ki = 47 nM T16691 C0LZ2J 46220503 Ki = 0.1995 nM T16691 CZJH90 46224877 IC50 = 5730 nM T16691 CFL32X 46224878 IC50 = 2580 nM T16691 C5FQ4S 46224879 Ki = 0.6166 nM T16691 CB0OH9 46224880 IC50 = 1680 nM T16691 C37TXV 46224881 IC50 = 910 nM T16691 CQ8P2A 46224914 IC50 = 180 nM T16691 C5DV2F 46224915 IC50 = 2810 nM T16691 CS0D4H 46224916 IC50 = 550 nM T16691 CC29VZ 46224917 IC50 = 1000 nM T16691 CH43AW 46224918 IC50 = 1750 nM T16691 C2G4FT 46224941 IC50 = 1440 nM T16691 CZX2L5 46224942 IC50 = 2950 nM T16691 C67UFY 46224943 IC50 = 5580 nM T16691 CUW7O3 46224944 IC50 = 1500 nM T16691 C4E6CK 46224945 IC50 = 1980 nM T16691 CW3R4Q 46224973 IC50 = 3720 nM T16691 CAZX21 46225000 IC50 = 692 nM T16691 CDR41P 46225001 IC50 = 1130 nM T16691 CDBP61 46225002 IC50 = 20700 nM T16691 C38OVM 46225027 IC50 = 2350 nM T16691 CFV3D0 46227395 Ki = 0.4 nM T16691 CY82LR 46227396 Ki = 3 nM T16691 C79UFN 46227404 Ki = 10 nM T16691 C42SVX 46700866 IC50 > 10000 nM T16691 CD0K6E 46700867 IC50 = 5000 nM T16691 CA4HD5 46830134 Ki = 0.68 nM T16691 C5TC2S 46830335 IC50 > 10000 nM T16691 C1K7FL 46830336 IC50 > 10000 nM T16691 C1N4KX 46842383 IC50 > 10000 nM T16691 CC62SX 46866711 IC50 = 16 nM T16691 C0HCI4 46867519 Ki = 0.499 nM T16691 C2B1NM 46867521 Ki = 0.256 nM T16691 C7K5AG 46867523 Ki = 28.8 nM T16691 CSLN36 46867524 Ki = 25.5 nM T16691 CCJ72Y 46867654 Ki = 869 nM T16691 C0HP4U 46867655 Ki = 1764 nM T16691 CRHN02 46880486 Ki = 6 nM T16691 C1T3YB 46880529 Ki = 10.7 nM T16691 CQC7S6 46880530 Ki = 68 nM T16691 CWI3U0 46880531 Ki = 16 nM T16691 C3HFU0 46880532 Ki = 4 nM T16691 CFK3A1 46880533 Ki = 21 nM T16691 CC9EQ0 46880606 Ki = 7.1 nM T16691 C6DO1B 46880607 Ki = 5.6 nM T16691 CZ4OL7 46880608 Ki = 4.7 nM T16691 CR8WY3 46880655 Ki = 3.5 nM T16691 CRZ1S3 46880656 Ki = 18 nM T16691 C47GTW 46880657 Ki = 9.6 nM T16691 C30YQL 46880658 Ki = 5 nM T16691 CCV2U9 46880659 Ki = 18 nM T16691 CFN34C 46880705 Ki = 15 nM T16691 C4RL1V 46880706 Ki = 72 nM T16691 CC8PU0 46880707 Ki = 3.2 nM T16691 CS7NP1 46880708 Ki = 1.3 nM T16691 CW5Y1T 46880709 Ki = 4.6 nM T16691 CW8DH2 46880756 Ki = 23.3 nM T16691 CM53AL 46880757 Ki = 6 nM T16691 C6FZG0 46880758 Ki = 1.5 nM T16691 C9JR7V 46880759 Ki = 2.8 nM T16691 CF8IJ2 46882520 Ki = 6.31 nM T16691 CQN87I 46882521 Ki = 125.89 nM T16691 C56ULO 46882522 Ki = 199.53 nM T16691 CX72IN 46882583 Ki = 15.85 nM T16691 C04JRH 46884709 Ki = 7.97 nM T16691 CB8GE1 46884818 IC50 > 10000 nM T16691 C4MQ0A 46884856 IC50 > 10000 nM T16691 CCNT25 46884898 IC50 > 10000 nM T16691 C3MSG2 46885027 IC50 > 10000 nM T16691 CB7XI0 46885213 IC50 = 3600 nM T16691 C8XK4D 46889325 Ki = 0.7943 nM T16691 CZK2Y7 46889326 Ki = 0.05012 nM T16691 C1NRH4 46889327 Ki = 5.012 nM T16691 CMF2K4 46889328 Ki = 0.1 nM T16691 CI0LR5 46889329 Ki = 1.259 nM T16691 CS86BA 46889349 Ki = 1 nM T16691 C8WJ7D 46889350 Ki = 0.1259 nM T16691 C6L0RO 46889351 Ki = 0.2512 nM T16691 CFCL20 46889352 Ki = 1.259 nM T16691 CI8OB1 46889353 Ki = 0.3162 nM T16691 C01JSO 46889472 Ki = 0.85 nM T16691 CUE0M9 46889856 Ki = 0.0631 nM T16691 CX7KU0 46889857 Ki = 25.12 nM T16691 CVKR52 46889858 Ki = 0.631 nM T16691 C04LNT 46889890 Ki = 0.1585 nM T16691 C2RL9U 46889891 Ki = 0.2512 nM T16691 C8AO0P 46889892 Ki = 0.3981 nM T16691 CA82ZW 46889893 Ki = 0.07943 nM T16691 CR13XZ 46889894 Ki = 3.981 nM T16691 CYU82R 46889895 Ki = 0.5012 nM T16691 CJRE76 46889915 Ki = 158.49 nM T16691 C4W2VY 46889916 Ki > 1000 nM T16691 CS8VY2 46889917 Ki = 0.3162 nM T16691 CV9ZF7 46889918 Ki = 0.1585 nM T16691 C81CYN 46889919 Ki = 7.943 nM T16691 CZY21R 46889920 Ki = 1.995 nM T16691 CC26DS 46890056 Ki = 31.62 nM T16691 C02CYN 46890057 Ki = 7.943 nM T16691 C9R5DS 46890058 Ki = 25.12 nM T16691 C63WEI 46890059 Ki = 50.12 nM T16691 C0FDW6 46890103 Ki = 158.49 nM T16691 C8BVJ4 46890104 Ki = 79.43 nM T16691 CWP20Q 46890105 Ki = 7.943 nM T16691 CGS9H6 46890106 Ki = 63.1 nM T16691 CDQS62 46890155 Ki = 0.3981 nM T16691 C3CX6A 46890156 Ki = 0.631 nM T16691 C9BUE2 46890157 Ki = 0.3981 nM T16691 CGB3Q0 46890158 Ki = 2.512 nM T16691 CO0GK6 46890188 Ki = 39.81 nM T16691 C1B8FI 46890189 Ki = 1.585 nM T16691 C5AGP8 46890190 Ki = 0.1259 nM T16691 CUC1W9 46890191 Ki = 1.585 nM T16691 C61GYF 46890192 Ki = 0.1 nM T16691 CKX3H2 46890218 Ki = 0.7943 nM T16691 C9M6BC 46890219 Ki = 3.981 nM T16691 CQE27V 46890220 Ki = 1.995 nM T16691 C6ZW7P 46890221 Ki = 0.3981 nM T16691 C1VND9 46890263 Ki = 31.62 nM T16691 CB5YT0 46890264 Ki = 0.1259 nM T16691 CE65DF 46890265 Ki = 3.981 nM T16691 C1CS6T 46890266 Ki = 1 nM T16691 CMVY84 46890267 Ki = 1.995 nM T16691 C75QXU 46890292 Ki = 31.62 nM T16691 C78KYS 46890293 Ki = 5.012 nM T16691 CO84JE 46890294 Ki = 15.85 nM T16691 CY42MI 46890295 Ki = 0.631 nM T16691 CL0Y8V 46890322 Ki = 0.1 nM T16691 CD8P6A 46890323 Ki = 6.31 nM T16691 C5QSL3 46890324 Ki = 0.1585 nM T16691 C9P5ZH 46890325 Ki = 0.1995 nM T16691 C50TPC 46890326 Ki = 0.2512 nM T16691 C4OBP5 46890884 Ki = 0.1585 nM T16691 C2Q1CG 46890885 Ki = 1.259 nM T16691 CAEV87 46890886 Ki = 19.95 nM T16691 CT71MK 46890887 Ki = 79.43 nM T16691 CHGA24 46890946 Ki = 31.62 nM T16691 CQSK68 46890947 Ki = 79.43 nM T16691 C4DMB0 46890948 Ki = 5.012 nM T16691 CRX51I 46890949 Ki = 31.62 nM T16691 C0ZN6Q 46891004 Ki = 25.12 nM T16691 CW6R3C 46891005 Ki = 31.62 nM T16691 CXRO49 46891006 Ki = 50.12 nM T16691 C72HAI 46891007 Ki = 316.23 nM T16691 CN9E0A 46891053 Ki = 125.89 nM T16691 C0JTL3 46891054 Ki = 63.1 nM T16691 CHZ25O 46891055 Ki = 316.23 nM T16691 CEH9I0 46891056 Ki = 316.23 nM T16691 C64NDL 46891111 Ki = 25.12 nM T16691 CI43LK 46891112 Ki = 19.95 nM T16691 CFC7A4 46891113 Ki = 25.12 nM T16691 CY0NP6 46891114 Ki = 100 nM T16691 C5ND3Q 46891174 Ki = 100 nM T16691 CRL43U 46891175 Ki = 125.89 nM T16691 CKB43Z 46891176 Ki = 31.62 nM T16691 CH86DQ 46933237 Ki = 23 nM T16691 CUTX67 46934428 IC50 = 3 nM T16691 CLT9W7 49780170 Ki = 447 nM T16691 CM98BZ 49780586 Ki = 27 nM T16691 CMA5Q3 49781032 Ki = 747 nM T16691 CS0EZ3 49781034 Ki = 215 nM T16691 CNR45W 49781036 Ki = 741 nM T16691 C1M7UP 49781038 Ki = 8 nM T16691 CL4R1V 49781250 Ki = 135 nM T16691 CMHL69 49781252 Ki = 175 nM T16691 CH1W6B 49781254 Ki = 554 nM T16691 C1QRV6 49781469 Ki = 194 nM T16691 C5X0JU 49781471 Ki = 523 nM T16691 CFSO43 49782361 Ki = 165 nM T16691 CQ39JR 49782362 Ki = 266 nM T16691 C2LZJ0 49783209 Ki = 489 nM T16691 C57SMG 49783415 Ki > 10000 nM T16691 C0TG6I 49783419 Ki > 10000 nM T16691 CB63SX 49798858 IC50 > 5000 nM T16691 C34YMO 49798859 IC50 = 120 nM T16691 C1RY7B 49799629 IC50 > 300 nM T16691 CHWT97 49799645 IC50 = 2260 nM T16691 CYC36S 49799656 IC50 = 580 nM T16691 CY4ZF0 49799663 IC50 = 1990 nM T16691 CPW4R7 49799664 IC50 = 1340 nM T16691 CAI82J 49799665 IC50 > 300 nM T16691 CL74MS 49799667 Ki = 14.7 nM T16691 CEJ4N3 49799678 IC50 > 300 nM T16691 COIW10 49799683 IC50 > 30 nM T16691 CG2W7R 49799684 IC50 > 30 nM T16691 C8AXI7 49799685 Ki = 26.3 nM T16691 C5AWK0 49799703 Ki = 103 nM T16691 CR40BA 49836386 IC50 = 37 nM T16691 C6N1PQ 49836504 Ki = 134 nM T16691 C1GJ9H 49836505 Ki = 125 nM T16691 CF98HT 49836507 Ki = 88 nM T16691 CSP1K6 49836508 Ki = 5.5 nM T16691 C6L8IS 49836509 Ki = 1.7 nM T16691 CU2X8O 49836615 Ki = 4 nM T16691 CI35ZA 49836616 Ki = 1 nM T16691 C2Z0KC 49836617 Ki = 8.1 nM T16691 C7F1MN 49836618 Ki = 1.1 nM T16691 CV3M8N 49836619 Ki = 12 nM T16691 C5HK3L 49836620 Ki = 0.9 nM T16691 C2SF3J 49836715 Ki = 7.8 nM T16691 C9NA6O 49836716 Ki = 2.6 nM T16691 C5T8CJ 49836717 Ki = 11 nM T16691 C6CZ9E 49836718 Ki = 110 nM T16691 CQ28NW 49836720 Ki = 124 nM T16691 CF71YC 49836721 Ki = 207 nM T16691 C7QAT9 49836823 Ki = 4.6 nM T16691 CJE9R5 49836824 Ki = 2.9 nM T16691 C8OAJ4 49836825 Ki = 1.7 nM T16691 C7G1VL 49836826 Ki = 1.7 nM T16691 CRUP23 49836827 Ki = 1.8 nM T16691 C36URZ 49836828 Ki = 1.8 nM T16691 C3DR7S 49836923 Ki = 1.4 nM T16691 C5DLH2 49836924 Ki = 2 nM T16691 C06HID 49836925 Ki = 22 nM T16691 C4R2YS 49850567 Ki = 794.33 nM T16691 C07JTU 49850570 Ki > 6309.57 nM T16691 CK68QR 49850672 Ki > 1584.89 nM T16691 CN5XR1 49850772 Ki > 10000 nM T16691 CR4EZ0 49850870 Ki > 2511.89 nM T16691 C5K4EC 49850872 Ki > 3981.07 nM T16691 C8AW0R 49850874 Ki > 1000 nM T16691 C9KIU1 49864289 IC50 = 6 nM T16691 CHO9C0 49864292 IC50 = 3 nM T16691 CU0TJ6 49864530 IC50 = 2191 nM T16691 C9FD2E 49864599 IC50 = 27 nM T16691 CVY4O3 49864600 IC50 = 422 nM T16691 CJF6T5 49864601 IC50 = 1180 nM T16691 C90MTG 49864602 IC50 = 644 nM T16691 C5BCS4 49864722 IC50 = 7 nM T16691 CKZO79 49864723 IC50 = 4 nM T16691 C74LZS 49864724 IC50 = 3 nM T16691 C2RY0J 50878551 Ki = 84 nM T16691 C1W6TV 50898777 Ki > 10000 nM T16691 CXMZ73 50898778 Ki > 10000 nM T16691 C8TA1J 51003550 IC50 = 28 nM T16691 CQ1UJ7 51003551 IC50 = 8 nM T16691 CGMI37 51003586 IC50 = 9 nM T16691 CE4KP1 51050257 Ki > 10000 nM T16691 C1DSG2 52912973 Ki = 8.2 nM T16691 CMJ5W7 52912975 Ki = 60 nM T16691 C2SCZ1 52913102 Ki = 4.1 nM T16691 C4JCT8 52913104 Ki = 1.8 nM T16691 C96RXD 52913108 Ki = 1.5 nM T16691 CPWJ93 52913218 Ki = 7.2 nM T16691 C0HSY1 52913224 Ki = 11 nM T16691 CF84CP 52913226 Ki = 35 nM T16691 C9HLS4 52913228 Ki = 6.3 nM T16691 CPFA98 52914691 Ki = 0.28 nM T16691 C1DQA4 52915868 Ki = 68.4 nM T16691 CBJS54 52915869 Ki = 2600 nM T16691 CB3UK9 52915979 Ki = 764 nM T16691 CZ2JV5 52915980 Ki = 489 nM T16691 CKA21J 52915982 Ki = 2200 nM T16691 C6G2KC 52915983 Ki = 1380 nM T16691 CL8C4Z 52915984 Ki = 2960 nM T16691 CRW65Z 52918030 Ki = 2.138 nM T16691 CP5LJ0 52918031 Ki = 7.586 nM T16691 CT8XL4 52918032 Ki = 0.2692 nM T16691 CYJM62 52940867 Ki = 1.698 nM T16691 CRI12K 52942395 Ki = 16 nM T16691 C08VZD 52945114 Ki = 90 nM T16691 C0UH4W 52945634 Ki = 1.413 nM T16691 C4PY3N 52945783 Ki = 0.7079 nM T16691 C9N6JV 52946845 Ki = 1 nM T16691 CA6H5W 52946846 Ki = 0.7943 nM T16691 CW0M1K 53259021 Ki = 2.9 nM T16691 CW2LS0 53303985 Ki = 0.75 nM T16691 CY92LZ 53310757 Ki = 10 nM T16691 C7GO1V 53316820 Ki = 3.4 nM T16691 C74VWQ 53316984 Ki = 0.5623 nM T16691 CK67HM 53317295 Ki = 30.2 nM T16691 CD1NU6 53317398 IC50 = 47 nM T16691 C02MWG 53318109 Ki = 1.4 nM T16691 C7V0JR 53318111 Ki = 12 nM T16691 CZP8O0 53318142 Ki = 24 nM T16691 C39KVU 53318267 Ki = 37.15 nM T16691 CY21CF 53318300 Ki = 114.82 nM T16691 C9ERL2 53318694 IC50 = 15 nM T16691 C2TI4Y 53319229 IC50 = 129 nM T16691 CLX9O5 53319441 Ki = 2.8 nM T16691 CI2M1K 53319443 Ki = 17 nM T16691 C5ZD7H 53319475 Ki = 44 nM T16691 C2VS1D 53319627 Ki = 7.943 nM T16691 CU6C0J 53319628 Ki = 3.89 nM T16691 CB3H8N 53319629 Ki = 9.55 nM T16691 C61DNP 53320009 IC50 = 26 nM T16691 C9ZDR5 53320010 IC50 = 61 nM T16691 CP6JY7 53320011 IC50 = 42 nM T16691 C8L9UI 53320746 Ki = 17 nM T16691 C8XA1F 53320775 Ki = 2.9 nM T16691 CKO65P 53320926 Ki = 3.236 nM T16691 CI5X2B 53320927 Ki = 15.14 nM T16691 CH5MP9 53320928 Ki = 37.15 nM T16691 C8HIW1 53320929 Ki = 1.995 nM T16691 CG98LC 53321318 IC50 = 165 nM T16691 C95JEG 53321319 IC50 = 58 nM T16691 C1EDO9 53322082 Ki = 24 nM T16691 CT34MP 53322258 Ki = 0.2818 nM T16691 CXR3D2 53322259 Ki = 3.162 nM T16691 C2Q5BC 53322547 Ki = 15.9 nM T16691 C5E6PM 53322548 Ki = 7.8 nM T16691 CME93W 53322637 IC50 = 353 nM T16691 CQLK01 53322638 IC50 = 11 nM T16691 C8FET1 53322935 Ki = 1.175 nM T16691 CG05WD 53323402 Ki = 0.24 nM T16691 CI1E4P 53323436 Ki = 12 nM T16691 CW8E9X 53323439 Ki = 4.8 nM T16691 CWP1D3 53323441 Ki = 107 nM T16691 CDV8Y5 53323599 Ki = 131.83 nM T16691 CCWQ31 53323600 Ki = 44.67 nM T16691 C1COV0 53323601 Ki = 11.75 nM T16691 C3I0AS 53323873 Ki = 25.5 nM T16691 C29PDB 53323972 IC50 = 17 nM T16691 C32YWL 53324045 Ki = 1695 nM T16691 CR4W9L 53324553 Ki > 10000 nM T16691 CG46AB 53324895 Ki = 154.88 nM T16691 C5WA0M 53324896 Ki = 1.445 nM T16691 C5BO0F 53324933 Ki = 22.91 nM T16691 CBHG43 53325160 Ki = 23.2 nM T16691 CRQF15 53325242 Ki = 1671 nM T16691 CNWH58 53325265 IC50 = 43 nM T16691 CKTW17 53325266 IC50 = 419 nM T16691 C4BM0X 53325267 IC50 = 7 nM T16691 CCE93D 53325519 Ki = 3.981 nM T16691 C0LRC8 53325577 Ki = 27 nM T16691 C87RZQ 53326022 Ki = 14 nM T16691 CMO38N 53326048 Ki = 65 nM T16691 C3G4ZS 53326175 Ki = 3.802 nM T16691 CNS74M 53326176 Ki = 0.2399 nM T16691 C5F2MI 53326177 Ki = 0.4786 nM T16691 CE6KO2 53326178 Ki = 0.6026 nM T16691 CTD50L 53326548 IC50 = 311 nM T16691 C7J8ZY 53327611 Ki = 4.4 nM T16691 C3MEG7 53327952 Ki = 8.913 nM T16691 CZL9W7 53327953 Ki = 95.5 nM T16691 CCL48Y 53327973 Ki = 20.89 nM T16691 CT5MJ8 53327974 Ki = 23.99 nM T16691 C5J8IG 53327976 Ki = 28.84 nM T16691 CGV7O2 53327979 Ki = 181.97 nM T16691 C4G7RQ 53327999 Ki = 25.7 nM T16691 CU9ON5 53328000 Ki = 23.99 nM T16691 C1HU7Y 53328001 Ki = 168 nM T16691 CD8C0G 54238415 Ki = 2039 nM T16691 C5Z1LN 54579956 IC50 = 2980 nM T16691 C8BSR5 54579957 IC50 = 8910 nM T16691 C9JZ7K 54580137 Ki = 300 nM T16691 CQKO51 54580394 Ki = 123 nM T16691 CYTC09 54580442 Ki = 5.72 nM T16691 CJO04Z 54580942 IC50 = 3240 nM T16691 CTN1V9 54580943 IC50 > 10000 nM T16691 CSK36H 54581122 Ki = 760 nM T16691 C43JTB 54581997 IC50 = 4340 nM T16691 CZ90MU 54581998 IC50 = 43200 nM T16691 CWB48T 54582158 Ki = 110 nM T16691 C5VS4M 54582159 Ki = 160 nM T16691 C8JG0O 54582465 Ki > 1000 nM T16691 CWY0J9 54582938 IC50 = 8360 nM T16691 CGZ2A0 54582939 IC50 = 1040 nM T16691 C63EMH 54582940 IC50 = 1590 nM T16691 C8QLJ2 54583109 Ki = 50 nM T16691 CE2SJ4 54583938 IC50 = 2060 nM T16691 CU2VZ8 54584108 Ki = 81 nM T16691 C2TE0Z 54584885 IC50 = 5800 nM T16691 CCN6S2 54585045 Ki = 78 nM T16691 CM56LK 54585846 IC50 = 10690 nM T16691 CNU5D7 54585847 IC50 = 6400 nM T16691 C03QMG 54585848 IC50 = 7470 nM T16691 C2SDF5 54586019 Ki = 110 nM T16691 COJ5R8 54586020 Ki = 330 nM T16691 C5QTZ6 54586316 Ki > 1000 nM T16691 C39KWS 54586812 IC50 = 15750 nM T16691 CY0G9U 54586813 IC50 > 10000 nM T16691 C4VA8X 54586997 Ki = 150 nM T16691 CD97AP 54752954 Ki = 4.8 nM T16691 CAZ5T6 54764323 Ki = 1950 nM T16691 COZ82F 55479093 Ki = 862 nM T16691 CN5M4X 56593642 Ki = 21.9 nM T16691 CIHK28 56593643 Ki = 119.4 nM T16691 C6B4VJ 56593644 Ki = 196.7 nM T16691 C1HEY6 56593645 Ki = 2.7 nM T16691 CWB5U7 56593646 Ki = 5.6 nM T16691 CL5G1M 56593647 Ki = 17.2 nM T16691 CX3Z4Q 56593797 Ki = 7.9 nM T16691 C3I1DH 56593798 Ki = 4.1 nM T16691 CE0GS3 56593799 Ki = 510.1 nM T16691 CND64S 56593800 Ki < 6 nM T16691 CXS0Y9 56593803 Ki = 49.9 nM T16691 CS7IL1 56593931 Ki = 6.4 nM T16691 C1LZQ6 56593932 Ki = 5.2 nM T16691 C1SUQ3 56593933 Ki = 71.1 nM T16691 C8WHT5 56593934 Ki = 7.2 nM T16691 CA4L8Y 56593935 Ki = 92 nM T16691 CN1QP8 56593936 Ki = 146.6 nM T16691 C4B6PY 56595280 Ki = 33.9 nM T16691 CW89BT 56595402 Ki = 2.8 nM T16691 C93KHG 56595403 Ki = 14.6 nM T16691 CK7F3O 56595404 Ki = 17.8 nM T16691 CE6YT2 56595405 Ki = 24.2 nM T16691 C9YF4L 56595406 Ki = 8 nM T16691 C3H8ED 56595407 Ki = 33.9 nM T16691 C1KA4D 56595408 Ki = 231.1 nM T16691 CDJ2H6 56595409 Ki > 1000 nM T16691 C4C3XQ 56595529 Ki = 23.9 nM T16691 C98WJL 56595531 Ki = 9.3 nM T16691 C42VXP 56595532 Ki > 1000 nM T16691 C14YAC 56595533 Ki = 321.8 nM T16691 C6KMX2 56595534 Ki = 8.2 nM T16691 CF41OI 56595535 Ki = 138.1 nM T16691 CHSO06 56595666 Ki = 18.5 nM T16691 CTXE98 56595667 Ki = 17 nM T16691 CI3V6E 56595668 Ki = 17.9 nM T16691 C6QL1G 56595669 Ki = 27.4 nM T16691 CSV45G 56595670 Ki = 26.6 nM T16691 CQ29HL 56595671 Ki = 7.9 nM T16691 CGK09C 56655504 Ki = 0.302 nM T16691 CM81NH 56655505 Ki = 0.9772 nM T16691 C3XC0S 56665086 Ki = 8.5 nM T16691 C8IE6A 56849575 Ki = 0.2188 nM T16691 C52SBY 56849576 Ki = 0.14 nM T16691 C1SH7I 56849577 Ki = 18.62 nM T16691 CO5T1U 56849578 Ki = 0.5754 nM T16691 C19QNC 56849579 Ki = 0.3467 nM T16691 C7U2DH 56849580 Ki = 69.18 nM T16691 CGDA95 56849581 Ki = 22.39 nM T16691 CN1PJ7 56849713 Ki = 112 nM T16691 CK1X6T 56849714 Ki = 16.6 nM T16691 CUF7Y5 56849715 Ki = 4.365 nM T16691 C9DX8R 56849716 Ki = 1.862 nM T16691 CN4A2H 56849717 Ki = 1.82 nM T16691 C4K3XA 56849719 Ki = 3.09 nM T16691 C16PYF 56849720 Ki = 33.88 nM T16691 C2E7OX 56849856 Ki = 4.677 nM T16691 C6QYO3 56849857 Ki = 0.8913 nM T16691 C1ZG7A 56933434 Ki = 13 nM T16691 CO0N2W 56943599 Ki = 18 nM T16691 C3DF5Z 56943600 Ki = 2.4 nM T16691 C19BDH 56943695 Ki = 25 nM T16691 CS7K3T 56943891 Ki = 71 nM T16691 CZ4L3S 56944082 Ki = 27 nM T16691 C5NI3K 56944086 Ki = 5200 nM T16691 C37BYO 56944186 Ki = 46 nM T16691 C9UOZ6 56944189 Ki = 95 nM T16691 CH7V9J 56944190 Ki = 26 nM T16691 CE49MC 56944191 Ki = 48 nM T16691 CX2RP5 56944287 Ki = 23 nM T16691 CB0P9N 56944383 Ki = 4.1 nM T16691 CEQ7I3 56944384 Ki = 3.3 nM T16691 CHWI01 56944473 Ki = 70 nM T16691 C6Y4ZQ 56944564 Ki = 5 nM T16691 C3B0MZ 56944565 Ki = 100 nM T16691 CI4KW0 56944664 Ki = 87 nM T16691 C39YHD 56944665 Ki = 8.8 nM T16691 C1W3GL 56944666 Ki = 2.4 nM T16691 C7J4UT 56944667 Ki = 140 nM T16691 CZT80U 56944668 Ki = 32 nM T16691 CTW2F5 56944763 Ki = 133 nM T16691 C50WEX 56944764 Ki = 210 nM T16691 CX0ZW2 56944859 Ki = 250 nM T16691 C1ST9U 56944860 Ki = 130 nM T16691 CQKL90 56944861 Ki = 100 nM T16691 CS5J6Y 56944862 Ki = 150 nM T16691 CFLB40 56944863 Ki = 110 nM T16691 C53OTR 56944864 Ki = 210 nM T16691 C5T3RI 56944951 Ki = 280 nM T16691 CR6H7U 56944952 Ki = 92 nM T16691 C1Y2RP 56944953 Ki = 180 nM T16691 C1BH7I 56944954 Ki = 30 nM T16691 CTK9I8 56944955 Ki = 46 nM T16691 CCF1A5 56944956 Ki = 10 nM T16691 C2YVT8 56945042 Ki = 35 nM T16691 CNI2G3 56945043 Ki = 10 nM T16691 CF9V3Q 56945045 Ki = 61 nM T16691 CE4S5M 56945046 Ki = 100 nM T16691 CHN2F6 56949640 Ki > 10000 nM T16691 CP31JY 56963265 Ki < 10 nM T16691 C1TC7Q 56963799 Ki > 10000 nM T16691 C3ZG6J 57325520 Ki = 139 nM T16691 CDK7B0 57325521 Ki = 16650 nM T16691 C3V5EM 57334669 Ki < 20 nM T16691 CSU54I 57334813 Ki < 100 nM T16691 C1PDV8 57334815 Ki < 10 nM T16691 C6VP7I 57334817 Ki < 10 nM T16691 CFNG46 57334819 Ki < 10 nM T16691 CJ23AC 57334821 Ki < 10 nM T16691 CX1AB6 57334823 Ki < 100 nM T16691 C2IY4K 57334968 Ki < 10 nM T16691 C0KP6N 57334970 Ki < 100 nM T16691 CU19GD 57334972 Ki < 10 nM T16691 CIJ0G1 57334974 Ki < 10 nM T16691 CS2O8K 57334976 Ki < 10 nM T16691 CX9W4N 57334978 Ki < 10 nM T16691 C4D6VQ 57335122 Ki < 10 nM T16691 CYS80P 57335124 Ki < 20 nM T16691 CZV73L 57335126 Ki < 100 nM T16691 CIQ08T 57335128 Ki < 100 nM T16691 CR9MZ4 57384073 Ki = 3567 nM T16691 C3HG2F 57390799 Ki = 1010 nM T16691 C83GWU 57391158 Ki = 6548 nM T16691 CS54WD 57391567 Ki = 11 nM T16691 CDL1T9 57391569 Ki = 21 nM T16691 CYD8T2 57391618 Ki = 11 nM T16691 CM8FX7 57391620 Ki = 562 nM T16691 CPE8N4 57391622 Ki = 750 nM T16691 CHG51U 57391624 Ki = 127 nM T16691 C78TOG 57391669 Ki = 49 nM T16691 CJP14X 57391729 Ki = 7.7 nM T16691 CZ28FL 57392612 Ki = 350 nM T16691 CO74HK 57392613 Ki = 4.8 nM T16691 C8OM2N 57392614 Ki = 51 nM T16691 CK89TZ 57392615 Ki = 32 nM T16691 C41ZCO 57393363 Ki = 11 nM T16691 CFI39D 57393365 Ki = 28 nM T16691 C6SO4I 57393467 Ki = 17.5 nM T16691 CJTY79 57393468 Ki = 2.1 nM T16691 CUF40C 57393877 Ki = 2652 nM T16691 CPU53I 57394331 Ki = 7.8 nM T16691 CFRN89 57394332 Ki = 192 nM T16691 CRQ16C 57394333 Ki = 0.74 nM T16691 C3S4KL 57394334 Ki = 0.28 nM T16691 C7VFQ3 57394663 Ki = 147 nM T16691 CN39YP 57395082 Ki = 48 nM T16691 CEW0O4 57395084 Ki = 155 nM T16691 CL96RC 57395086 Ki = 3765 nM T16691 CTG35L 57395190 Ki = 139 nM T16691 CJ15YT 57395598 Ki = 590 nM T16691 C6V3GB 57396088 Ki = 156 nM T16691 C51GCK 57396417 Ki = 17150 nM T16691 CZ2SJ8 57396419 Ki = 24840 nM T16691 C6HBG0 57396813 Ki = 4 nM T16691 CKQH25 57396848 Ki = 32 nM T16691 C92SIX 57396850 Ki = 15 nM T16691 CZ8KA2 57396855 Ki = 1725 nM T16691 CN7QE4 57396857 Ki = 2209 nM T16691 C3L4ED 57396970 Ki = 1.6 nM T16691 CKM78R 57397900 Ki = 54 nM T16691 CYCN81 57397901 Ki > 10000 nM T16691 C51XVB 57398613 Ki = 83 nM T16691 CV1P0K 57398615 Ki = 17 nM T16691 C7W5XA 57398619 Ki = 2757 nM T16691 CY3D5F 57398717 Ki = 22 nM T16691 C2DRP9 57398718 Ki = 5.6 nM T16691 CMA0U2 57398803 Ki = 2.7 nM T16691 CTF76G 57399090 Ki = 825 nM T16691 C0XFB2 57399091 Ki = 2159 nM T16691 CI6ET3 57399092 Ki = 1920 nM T16691 CMX4K5 57399093 Ki = 4587 nM T16691 CR5WK3 57399547 Ki = 91 nM T16691 CUQ14N 57399548 Ki = 52 nM T16691 C3PZ2J 57399549 Ki = 4.6 nM T16691 CAN0W7 57399866 Ki = 10570 nM T16691 C9BG7C 57399868 Ki = 5043 nM T16691 CH0CL2 57400234 Ki = 2 nM T16691 CAI2N9 57400275 Ki = 2.9 nM T16691 CYKA35 57400277 Ki = 385 nM T16691 C5HGO2 57400281 Ki = 397 nM T16691 CWY4G5 57400391 Ki = 18 nM T16691 CQ9KY6 57400392 Ki = 22.3 nM T16691 C4IB3E 57400477 Ki = 46 nM T16691 CT7Q3E 57400828 Ki = 1082 nM T16691 C3D1UP 57400830 Ki = 14460 nM T16691 CC6BP9 57401298 Ki = 37 nM T16691 C5GPJ0 57401515 Ki = 29070 nM T16691 CG8MF3 57401516 Ki = 20410 nM T16691 CP6JM8 57402070 Ki = 38 nM T16691 C2GMY9 57402072 Ki = 203 nM T16691 C7CG1T 57402187 Ki = 16 nM T16691 CN9J5I 57402588 Ki = 1518 nM T16691 CTD09H 57403055 Ki = 814 nM T16691 C75RIG 57403056 Ki = 131 nM T16691 C75KOS 57403057 Ki = 0.68 nM T16691 C4CD2L 57403058 Ki = 0.81 nM T16691 CD2WK3 57403833 Ki = 37 nM T16691 CO24AV 57403835 Ki = 85 nM T16691 CIL3W4 57403837 Ki = 64 nM T16691 C3A1YW 57403839 Ki = 339 nM T16691 CA10YX 57403841 Ki = 1535 nM T16691 CP4OY8 57520121 IC50 = 360 nM T16691 CFW1T3 57520122 IC50 = 440 nM T16691 CQ7GV6 58149665 Ki = 7.7 nM T16691 CC79AK 58149671 Ki > 10000 nM T16691 CUI3O8 58149672 Ki = 35.7 nM T16691 C4Y5KG 58158668 Ki = 20.6 nM T16691 C7CN4T 58158673 Ki = 399.1 nM T16691 CVI3T6 58158682 Ki = 18.5 nM T16691 CRI13V 58158707 Ki = 28.6 nM T16691 C31CYM 58158709 Ki = 31.6 nM T16691 CP9A8Q 58158717 Ki = 160.2 nM T16691 CPME36 58158719 Ki = 14.6 nM T16691 C3VF9E 58158721 Ki = 1.8 nM T16691 C8EVD4 58158738 Ki = 14.2 nM T16691 CK10XC 58158739 Ki = 5.8 nM T16691 C2JP3M 58158748 Ki = 97.2 nM T16691 CN6K3Z 58158749 Ki = 6.1 nM T16691 CBH2G3 59017478 Ki = 1 nM T16691 CZ2E6P 59339309 Ki = 205.9 nM T16691 C2RFW6 59339335 Ki = 7.2 nM T16691 C93KWC 59339383 Ki = 8.7 nM T16691 CKI6R9 60141574 IC50 = 3600 nM T16691 C6AUO2 66800823 Ki = 120 nM T16691 C34ACQ 66800909 Ki = 27 nM T16691 CGT9E6 66800910 Ki = 130 nM T16691 C0QY7D 66800916 Ki = 54 nM T16691 CM58FG 66800926 Ki > 10000 nM T16691 CQ43WD 66800934 Ki = 47 nM T16691 CK0I5J 66800939 Ki = 40 nM T16691 C0X2SF 66800942 Ki = 430 nM T16691 CN30YT 66800947 Ki = 9.2 nM T16691 CZ3MR6 66800959 Ki = 34 nM T16691 C92CMO 66800965 Ki = 320 nM T16691 CFPK92 66800991 Ki = 84 nM T16691 C13GMO 66801000 Ki = 63 nM T16691 CZ1TF9 66801018 Ki = 17 nM T16691 CBO9U3 66801028 Ki = 35 nM T16691 C3K8DC 66801052 Ki = 300 nM T16691 CA4DM3 66801062 Ki = 40 nM T16691 C2OUX9 66801107 Ki = 22 nM T16691 C4J5RZ 66801115 Ki = 110 nM T16691 C1H8BS 66801116 Ki > 10000 nM T16691 C4JGC6 66801120 Ki = 26 nM T16691 CX2GN1 66801139 Ki = 13 nM T16691 C1NG8S 66801140 Ki = 53 nM T16691 CR7OW6 66801158 Ki = 6.2 nM T16691 CJU53X 66801160 Ki = 5.1 nM T16691 CH3BJ8 66801167 Ki = 83 nM T16691 C0AV5M 66801173 Ki = 33 nM T16691 C0V9EF 66801186 Ki = 100 nM T16691 CTHY41 66801210 Ki = 1.8 nM T16691 CSD67P 66801225 Ki = 13 nM T16691 C8J3YU 66801226 Ki = 330 nM T16691 CX45OZ 66801229 Ki = 680 nM T16691 C1S0EV 66801230 Ki = 42 nM T16691 C7S1KY 66801234 Ki = 1.6 nM T16691 CB53AV 66801246 Ki = 100 nM T16691 C3F1TZ 66801251 Ki = 44 nM T16691 CF8O9U 66801259 Ki > 10000 nM T16691 C2Q9FS 66801263 Ki = 29 nM T16691 C7Y9VP 66801267 Ki = 2300 nM T16691 CED17M 66801271 Ki = 66 nM T16691 C41VYW 66801295 Ki = 200 nM T16691 C2FYL1 66801333 Ki = 1100 nM T16691 CS75LK 66801335 Ki = 56 nM T16691 CR2N0J 66801344 Ki = 220 nM T16691 CDH7S9 66801346 Ki = 7.1 nM T16691 CGC4U6 66801354 Ki = 1600 nM T16691 CY4FM5 66801379 Ki = 120 nM T16691 C3RX4C 66801425 Ki = 250 nM T16691 C7JD0I 66801429 Ki = 130 nM T16691 CN8OU1 66801430 Ki = 100 nM T16691 C93EGP 66801455 Ki = 140 nM T16691 COR1H8 66801528 Ki = 67 nM T16691 C1F3YV 66801537 Ki = 20 nM T16691 CIRW86 66801551 Ki = 3.4 nM T16691 C75WXP 66801561 Ki = 200 nM T16691 C8H5PD 66801565 Ki = 23 nM T16691 CT5SP8 66801605 Ki = 45 nM T16691 C8MH0I 66801613 Ki = 15 nM T16691 CC8JV6 66801624 Ki = 180 nM T16691 C3EI2F 66801625 Ki = 350 nM T16691 C49XBJ 66801673 Ki = 1100 nM T16691 C0XG6B 66801701 Ki = 360 nM T16691 C42EBQ 66801837 Ki = 250 nM T16691 CW3AI2 66803474 Ki = 6.4 nM T16691 CPKH06 66803497 Ki = 120 nM T16691 CNJE57 66803500 Ki = 330 nM T16691 CN6FZ1 66803595 Ki = 3.5 nM T16691 CD7Y0H 66852770 Ki = 7.5 nM T16691 CR26JV 67156504 Ki = 5 nM T16691 C1LEH8 67268994 Ki = 248 nM T16691 CLK0B7 68014784 Ki = 48.3 nM T16691 CYHG09 68014793 Ki = 153 nM T16691 CLA7F3 68281136 Ki = 140 nM T16691 C84MZH 68281137 Ki = 4800 nM T16691 CDG8X3 68544797 Ki = 2.82 nM T16691 CV54LO 68638941 Ki = 23.5 nM T16691 CD3U6K 68731121 Ki > 10000 nM T16691 C6IP8Q 69082816 Ki > 10000 nM T16691 CH3A6M 69485025 Ki = 36.3 nM T16691 C9L0TF 70245924 Ki = 0.66 nM T16691 CTE40A 70301391 Ki = 0.93 nM T16691 CC43QK 71151588 Ki = 1 nM T16691 CG5A0O 71151591 Ki = 23 nM T16691 CB4K3V 71151664 Ki = 24 nM T16691 CO8CB3 71151683 Ki = 9.9 nM T16691 C5U2BI 71151704 Ki = 2.3 nM T16691 CU74VQ 71151756 Ki = 11 nM T16691 CVMJ59 71151757 Ki = 2.8 nM T16691 C4AF8X 71151767 Ki = 45 nM T16691 CN05SR 71151870 Ki = 83 nM T16691 CG18YE 71151889 Ki = 12.6 nM T16691 CC9M3F 71151924 Ki = 20 nM T16691 CP9A6W 71151925 Ki = 16 nM T16691 C2V5SX 71151929 Ki = 6.9 nM T16691 CM4QC9 71151933 Ki = 0.4 nM T16691 CYP91I 71151953 Ki = 7.3 nM T16691 CN4AJ3 71152026 Ki = 100 nM T16691 CZM5O9 71163244 Ki = 118 nM T16691 C91SZN 71449641 Ki = 315 nM T16691 C2GCN7 71449642 Ki = 957 nM T16691 CQN93U 71449643 Ki = 327 nM T16691 CEJ3B4 71449644 Ki = 156 nM T16691 C5SAJ1 71449645 Ki = 537 nM T16691 CLM07O 71449795 Ki = 2.85 nM T16691 CM0TQ2 71449796 Ki = 10.4 nM T16691 C6LD8A 71449798 Ki = 13.1 nM T16691 C3XNC2 71450247 Ki = 6256 nM T16691 CI95UR 71450930 Ki = 49 nM T16691 CHT21G 71451454 Ki = 2759 nM T16691 C2QZL4 71451455 Ki = 147 nM T16691 CXI5Q2 71451456 Ki = 3785 nM T16691 CKJZ57 71451457 Ki = 258 nM T16691 C0F1HU 71451458 Ki = 185 nM T16691 CTZ24N 71451459 Ki = 200 nM T16691 C70JUP 71451460 Ki = 202 nM T16691 C10IGU 71451603 Ki = 5.02 nM T16691 C8VXH9 71451605 Ki = 17.12 nM T16691 CYK20Z 71452384 Ki > 10000 nM T16691 CKI58Z 71453278 Ki = 1799 nM T16691 C1QM8D 71453279 Ki = 225 nM T16691 C6O4KT 71453280 Ki = 515 nM T16691 CL49VI 71453281 Ki = 245 nM T16691 CGXT64 71453282 Ki = 551 nM T16691 C65RKA 71453361 Ki = 73.4 nM T16691 CE0R9D 71454275 IC50 > 580000 nM T16691 CGO13Q 71454997 Ki = 410 nM T16691 C0K1JV 71454998 Ki = 177 nM T16691 C3JF1D 71454999 Ki = 240 nM T16691 C2QZ1N 71455000 Ki = 199 nM T16691 C6FE5D 71455001 Ki = 951 nM T16691 C4L0JN 71455002 Ki = 102 nM T16691 CTP83A 71455149 Ki = 4.3 nM T16691 CAQF34 71455625 Ki > 10000 nM T16691 CWR40I 71456780 Ki = 831 nM T16691 CZUX67 71456781 Ki = 267 nM T16691 CZ17FC 71456782 Ki = 248 nM T16691 CKF09U 71456783 Ki = 96 nM T16691 CJKV72 71456784 Ki = 271 nM T16691 C7C2ST 71456942 Ki = 3.63 nM T16691 C35RLC 71456943 Ki = 70.6 nM T16691 CQ6WA2 71456944 Ki = 61.21 nM T16691 CMJ1O9 71457409 Ki > 10000 nM T16691 C37EBC 71458647 Ki = 313 nM T16691 CM6OP1 71458648 Ki = 2124 nM T16691 CRGE05 71458649 Ki = 1779 nM T16691 CJN4S1 71458650 Ki = 91 nM T16691 CNT5J9 71458651 Ki = 504 nM T16691 C3NAM7 71458652 Ki = 357 nM T16691 CR9I8F 71458723 Ki = 39.1 nM T16691 C3RS9W 71458811 Ki = 1.6 nM T16691 CY05VS 71458812 Ki = 4.68 nM T16691 CS83IF 71459269 Ki > 10000 nM T16691 CK5T4P 71459604 Ki > 10000 nM T16691 CG0WO9 71459954 EC50 = 0.4 nM T16691 CT17XB 71460468 Ki = 1761 nM T16691 C63YLA 71461049 Ki > 10000 nM T16691 CJD96I 71461050 Ki > 10000 nM T16691 C7AX1Q 71462178 Ki = 1335 nM T16691 C1CS0Z 71462179 Ki = 102 nM T16691 CDX7M6 71462329 Ki = 5.01 nM T16691 CF15LQ 71462330 Ki = 9.15 nM T16691 C5KJZ7 71462331 Ki = 29.01 nM T16691 C4P3JU 71462776 Ki > 10000 nM T16691 C3GUQ2 71462777 Ki > 10000 nM T16691 CP2SY9 71463515 Ki = 100 nM T16691 CJYW50 71463516 Ki = 84 nM T16691 CB4K0Y 71463517 Ki = 41 nM T16691 CI98TK 71463518 Ki = 2600 nM T16691 CC2PE0 71463519 Ki = 270 nM T16691 CJ57BD 71463520 Ki = 4900 nM T16691 CG4AF3 71463521 Ki = 2900 nM T16691 C1E9HB 71502591 Ki = 13 nM T16691 CE9ZL1 71502631 Ki = 7.6 nM T16691 CQ3EZ2 71502632 Ki = 5.4 nM T16691 CQ8FW4 71502633 Ki = 1.7 nM T16691 CBY90L 71502676 Ki = 3.8 nM T16691 CT2ME3 71574204 Ki = 220 nM T16691 C3SXR5 71574206 Ki = 901 nM T16691 C2YRI9 71574208 Ki = 326 nM T16691 C62RWV 71574210 Ki = 257 nM T16691 CKC53S 71574212 Ki = 1331 nM T16691 CNV42M 71574298 Ki = 555 nM T16691 C9PGQ1 71574300 Ki = 484 nM T16691 C2LXH5 71574302 Ki = 301 nM T16691 C2YPB8 71574304 Ki = 598 nM T16691 CK7GM0 71574306 Ki = 454 nM T16691 C0W2YA 71727193 Ki = 9363 nM T16691 C79TLS 71727194 Ki = 19100 nM T16691 CFB10W 71727195 Ki = 8836 nM T16691 C6CIB5 71727196 Ki = 13600 nM T16691 C7Z3JS 71727308 Ki = 5939 nM T16691 C2W5JT 71727892 Ki = 0.16 nM T16691 CR4Q3A 71769065 IC50 = 1800 nM T16691 CGMN49 71769066 IC50 = 7400 nM T16691 CC07ST 71769190 IC50 = 2900 nM T16691 CFPC45 71769315 IC50 = 6600 nM T16691 C17QTG 71769424 IC50 = 1400 nM T16691 CIZ98N 71770821 IC50 = 2400 nM T16691 C0K8NC 71770822 IC50 = 4740 nM T16691 C6CVD5 71770944 IC50 = 2040 nM T16691 C9PIE1 71813685 IC50 = 5220 nM T16691 CH7IG2 71813833 IC50 = 3280 nM T16691 C0P6JL 71813835 IC50 = 6770 nM T16691 C0TMX6 71813838 IC50 = 1660 nM T16691 C1R0QA 71813986 IC50 = 580 nM T16691 C0A3SV 71813988 IC50 = 7080 nM T16691 C7VP8T 71814155 IC50 = 770 nM T16691 C7I9KL 71814157 IC50 = 310 nM T16691 CL4B0J 71814318 IC50 = 310 nM T16691 C53MXL 71815503 IC50 = 740 nM T16691 C3ATN5 72197484 IC50 = 36.8 nM T16691 C20HSN 72197485 IC50 = 22.2 nM T16691 CN8A5R 72197486 IC50 = 21.8 nM T16691 CL3BF7 72197668 IC50 = 30.4 nM T16691 CUVJ59 72197845 Ki = 63 nM T16691 CIKU20 72198011 Ki = 159 nM T16691 COH95V 72198014 Ki = 264 nM T16691 C0WY2V 72198191 Ki = 1146 nM T16691 CWH6T3 72548703 IC50 = 254 nM T16691 C80VRM 72549033 Ki = 0.22 nM T16691 C8Z0NM 72550642 Ki = 1517 nM T16691 CL6W2Q 72550645 Ki = 1321 nM T16691 C78LYM 72698087 Ki > 10000 nM T16691 C63HPK 72698088 Ki > 10000 nM T16691 CC6Q5R 72771081 Ki < 100 nM T16691 CC65OA 73213195 Ki = 273 nM T16691 CW83DK 73213196 Ki > 10000 nM T16691 CXM8O2 73347306 EC50 = 5.3 nM T16691 C9X8GY 73347307 EC50 = 32 nM T16691 CE2H9S 73347593 Ki = 8.3 nM T16691 CH9M8C 73347610 IC50 = 3600 nM T16691 CR97NO 73347825 Ki > 10000 nM T16691 CY60RD 73347826 Ki > 10000 nM T16691 C9ML2B 73348100 Ki = 12.5 nM T16691 C0V3YM 73349113 Ki = 30.1 nM T16691 CIJ64B 73349123 IC50 = 3800 nM T16691 CVUT85 73350387 EC50 = 6.6 nM T16691 C8GQK9 73350823 Ki = 187 nM T16691 CC8I7X 73351903 EC50 = 32 nM T16691 C0C7PV 73351904 IC50 = 100 nM T16691 CG4M8P 73351905 IC50 = 1000 nM T16691 C1YOX0 73351911 IC50 = 80 nM T16691 C0PT9Z 73353367 IC50 = 100 nM T16691 C89NZA 73353655 Ki = 1.65 nM T16691 CAR7Z5 73354882 EC50 = 2.7 nM T16691 CFI26G 73354883 IC50 = 9 nM T16691 C5N7EC 73356442 EC50 = 21 nM T16691 CET52A 73356443 IC50 = 700 nM T16691 CUB97Z 74538690 Ki = 830 nM T16691 COB03V 74763017 Ki = 15 nM T16691 C2E7QW 75201901 Ki = 8100 nM T16691 C8IDL3 75306277 Ki = 15.85 nM T16691 C45OSP 76284193 Ki = 2518 nM T16691 CIU19B 76328541 IC50 = 330 nM T16691 C9S0XK 86288947 Ki = 10790 nM T16691 CIA2B8 86294717 Ki = 14 nM T16691 CCY5N2 86302554 Ki = 2.6 nM T16691 CHE2U4 90178632 Ki = 148 nM T16691 C86OJA 90468813 Ki = 3 nM T16691 CFDW68 90644074 Ki = 1500 nM T16691 C0T8RE 90644075 Ki = 2200 nM T16691 C2KE9G 90644076 Ki > 10000 nM T16691 C1SOF5 90644077 Ki = 35 nM T16691 CIE9Z2 90644078 Ki = 560 nM T16691 CWMU25 90644511 IC50 = 280 nM T16691 CYB8K4 90644513 Ki = 46.77 nM T16691 C3U1IQ 90645147 Ki = 2707 nM T16691 CVG2C1 90654672 Ki = 282 nM T16691 CJG31T 90654831 Ki = 4139 nM T16691 CMU45O 90654832 Ki = 3071 nM T16691 C14NPE 90654833 Ki = 9600 nM T16691 C3C4BW 90654834 Ki = 25520 nM T16691 C8QWR3 90654835 Ki = 14650 nM T16691 C6ZR9L 90654837 Ki = 4368 nM T16691 C0AC7R 90654839 Ki = 8611 nM T16691 CKLG40 90654841 Ki = 2926 nM T16691 C5JS8D 90654843 Ki = 2506 nM T16691 C4VHZ6 90654845 Ki = 1945 nM T16691 CG78PS 90654847 Ki = 7469 nM T16691 CL39WP 90654849 Ki = 8104 nM T16691 C0TVQ9 90654851 Ki = 1762 nM T16691 C4I1CU 90654853 Ki = 395 nM T16691 CZ28YC 90654855 Ki = 314 nM T16691 CRO83N 90654857 Ki = 2879 nM T16691 CTN1D3 90656153 Ki = 54 nM T16691 C1I3ZB 90656154 Ki = 100 nM T16691 CE6C9U 90656155 Ki = 650 nM T16691 C1Z3PQ 90656156 Ki = 1200 nM T16691 CC95ZU 90656157 Ki = 140 nM T16691 CZ9OD5 90656158 Ki = 70 nM T16691 CIB5P7 90656159 Ki = 84 nM T16691 C30EKW 90656160 Ki = 48 nM T16691 C5TD0H 90656161 Ki = 4100 nM T16691 C6T8KC 90656162 Ki > 30000 nM T16691 CAOR80 90656163 Ki = 55 nM T16691 CN4VR5 90656164 Ki = 4900 nM T16691 CN5TQ9 90656165 Ki = 10 nM T16691 C6S7EM 90656166 Ki = 16 nM T16691 CG7IS2 90656167 Ki = 15 nM T16691 CPQ39B 90656168 Ki = 47 nM T16691 CF8M7I 90656169 Ki = 87 nM T16691 C23VSZ 90656170 Ki = 10 nM T16691 CX24VH 90656171 Ki = 240 nM T16691 CW07FN 90656172 Ki = 140 nM T16691 C5QK6I 90656173 Ki = 1900 nM T16691 C3S9CI 90656174 Ki = 150 nM T16691 CYW04S 90656175 Ki = 330 nM T16691 CCOV98 90664359 Ki = 19460 nM T16691 C4MUI2 90664601 IC50 = 136 nM T16691 CXD5Q9 90664621 Ki = 14420 nM T16691 CWNR05 90664684 IC50 = 780 nM T16691 CHT7D5 90664962 IC50 = 1682 nM T16691 CACG19 90666899 Ki = 213.8 nM T16691 CODM50 90666903 Ki = 354.81 nM T16691 CFEO02 91971999 IC50 = 0.17 nM T16691 CUQ6V0 92042918 Ki < 1000 nM T16691 CPEM50 118456745 IC50 = 2.7 nM T16691 CEMZ15 118464420 Ki = 3031 nM T16691 CV2L6O 118464425 Ki = 4777 nM T16691 CFNG86 118464427 Ki = 5909 nM T16691 C7AMX4 118464990 IC50 = 31 nM T16691 CJ6YV9 118464995 IC50 = 0.92 nM T16691 CNS8P6 118464996 IC50 = 0.5 nM T16691 CUDR52 118464997 IC50 = 1.3 nM T16691 C46JBK 118464998 IC50 = 1 nM T16691 C5MI2D 118465009 IC50 = 2 nM T16691 CYMK37 118465011 IC50 = 0.28 nM T16691 C2D0KT 118465015 IC50 = 3.2 nM T16691 CZ1NX5 118465021 IC50 = 5.5 nM T16691 C0VGE2 118465023 IC50 = 0.46 nM T16691 CU0I6P 118465024 IC50 = 11 nM T16691 CZD43F 118465025 IC50 = 1.6 nM T16691 CR38IZ 118465026 IC50 = 2.6 nM T16691 CG6N7X 118465027 IC50 = 4.1 nM T16691 C13GUZ 118465034 IC50 = 16 nM T16691 CO3W8Q 118465035 IC50 = 1.3 nM T16691 COKX07 118465038 IC50 = 11 nM T16691 CWR0B1 118465045 IC50 = 0.31 nM T16691 CAUL06 118465046 IC50 = 5 nM T16691 C98REJ 118465048 IC50 = 1.4 nM T16691 CKZ50J 118465050 IC50 = 1.7 nM T16691 CQ4RU0 118465051 IC50 = 2.1 nM T16691 CH4E0L 118465054 IC50 = 1.1 nM T16691 C7TEA2 118465055 IC50 = 3.7 nM T16691 C3VZ5N 118465064 IC50 = 1.2 nM T16691 C0TP5K 118465065 IC50 = 2.3 nM T16691 C10IRY 118465087 IC50 = 2.1 nM T16691 CJ29GH 118465171 IC50 = 0.69 nM T16691 CK04PJ 118512792 IC50 = 1420 nM T16691 CX71LC 118512797 IC50 = 10900 nM T16691 C76UQN 118512804 IC50 = 1780 nM T16691 CNE79I 118512805 IC50 = 3300 nM T16691 C78ZFD 118512807 IC50 = 8780 nM T16691 C3AK8G 118512815 IC50 = 2430 nM T16691 CA91YU 118512827 IC50 = 5650 nM T16691 CB5I1A 118512841 IC50 = 4010 nM T16691 CMSN80 118626035 Ki = 82 nM T16691 CT3AI0 118626042 Ki = 2057 nM T16691 CKNJ72 118626045 Ki = 72 nM T16691 CGB42Y 118626088 Ki = 996 nM T16691 C0XJT5 118626089 Ki = 116 nM T16691 CIE4C7 118626101 Ki = 766 nM T16691 C1NYS5 118626120 Ki = 1483 nM T16691 CPG04R 118626121 Ki = 9 nM T16691 C3S5LJ 118626129 Ki = 13 nM T16691 CY3F0N 118626140 Ki = 60 nM T16691 CE07IQ 118626142 Ki = 11 nM T16691 C72OZY 118626161 Ki = 38 nM T16691 CY3E7S 118626169 Ki = 1263 nM T16691 CHRB75 118626208 Ki = 2533 nM T16691 CIM3W2 118712402 Ki = 10 nM T16691 C5IF4Q 118712403 Ki = 99 nM T16691 C93OIS 118712404 Ki = 118 nM T16691 CHT8B0 118712405 Ki = 1 nM T16691 CKRA34 118712406 Ki = 11 nM T16691 C1JG4L 118712407 Ki = 1.2 nM T16691 C6XZC4 118712408 Ki = 3.8 nM T16691 CVL8B4 118712409 Ki = 0.9 nM T16691 C1F9ZM 118724639 Ki = 10350 nM T16691 CE05XG 118727442 IC50 = 1830 nM T16691 C1ZH2I 118727443 IC50 = 4970 nM T16691 C0M5AR 118727444 IC50 = 6340 nM T16691 CDHS51 118727445 IC50 = 2120 nM T16691 CWZ7P0 118727447 IC50 = 1400 nM T16691 CH9V1A 118727448 IC50 = 2440 nM T16691 C6AZG2 118727449 IC50 = 2960 nM T16691 CZ1LD0 118727450 IC50 = 2530 nM T16691 CB97QH 118727451 IC50 = 3900 nM T16691 C5O2NU 118729733 Ki = 5805 nM T16691 C8GKX6 118731351 Ki = 594 nM T16691 CQ8F6C 118731354 Ki = 603 nM T16691 CU12XM 118731356 Ki = 376 nM T16691 CD5RI3 118731502 Ki = 22 nM T16691 C5UQ3P 118731503 Ki = 52 nM T16691 CB6H8O 118731504 Ki = 150 nM T16691 CLFJ64 118731505 Ki = 140 nM T16691 CFPX32 118731506 Ki = 150 nM T16691 CL35UJ 118731507 Ki = 52 nM T16691 CF3TJ0 118731508 Ki = 590 nM T16691 CRBZ61 118731509 Ki = 33 nM T16691 CRJ4A6 118731510 Ki = 490 nM T16691 CCPL16 118731511 Ki = 57 nM T16691 C2POB0 118731512 Ki = 680 nM T16691 CZRB40 118731513 Ki = 62 nM T16691 CED26B 118732439 Ki = 100 nM T16691 C75OXS 118736395 Ki > 1000 nM T16691 C74FCM 118736396 Ki = 86 nM T16691 C3F8PA 118736397 Ki = 839 nM T16691 CWU1A0 121238068 Ki = 20 nM T16691 C8I7TE 121238069 Ki = 95 nM T16691 C5X8MN 122186880 Ki = 627 nM T16691 C7ODW3 122195524 Ki < 300 nM T16691 CBHT01 122377930 Ki = 471 nM T16691 CLW53P 122483274 Ki = 879 nM T16691 C4QM2E 124247485 Ki = 416 nM T16691 CVJR26 125513586 Ki = 450 nM T16691 CX1L8T 126720370 Ki = 165 nM T16691 C8Q3HT 126720389 Ki = 337 nM T16691 CLWM12 126720394 Ki = 7 nM T16691 CH98YW 126720395 Ki = 108 nM T16691 C8Q1JB 126720403 Ki = 13 nM T16691 CB3H1C 126720406 Ki = 165 nM T16691 CU3D1V 126720407 Ki = 92 nM T16691 CHCB04 126720410 Ki = 61 nM T16691 C02ZVU 126720412 Ki = 142 nM T16691 CEQ5C2 126720417 Ki = 21 nM T16691 C1U3SZ 126720425 Ki = 20 nM T16691 CWOK84 126720426 Ki = 57 nM T16691 CQ9Y8F 126720427 Ki = 162 nM T16691 C2QSR6 126720429 Ki = 101 nM T16691 C5G8FD 126720440 Ki = 6 nM T16691 C59SNQ 126720442 Ki = 107 nM T16691 CVL36P 126720443 Ki = 56 nM T16691 C2ZFI0 126720444 Ki = 42 nM T16691 CZN9Q7 126720445 Ki = 254 nM T16691 CT13NH 126720448 Ki = 177 nM T16691 CFG95T 126720449 Ki = 829 nM T16691 CIHZ54 127025242 Ki = 539 nM T16691 CCY7P3 127025243 Ki = 559 nM T16691 CTBN56 127026052 Ki = 74.13 nM T16691 CTYP30 127026133 Ki = 325 nM T16691 C0SZI4 127026515 Ki = 595 nM T16691 CX6EI2 127026750 Ki = 281 nM T16691 C8MC1I 127028408 Ki = 111 nM T16691 C6ARO4 127031618 Ki > 1000 nM T16691 CS16FX 127031619 Ki = 251.2 nM T16691 C34QDL 127032187 Ki = 210.2 nM T16691 C4V7RY 127032188 Ki > 1000 nM T16691 C3H2LU 127032424 Ki = 47.5 nM T16691 CJF14Z 127033666 Ki = 97.1 nM T16691 CZ61LK 127034966 EC50 > 5011.87 nM T16691 CA0SN5 127034967 EC50 > 5011.87 nM T16691 CU49VE 127036186 Ki = 741.31 nM T16691 CG06BD 127036932 Ki = 69.18 nM T16691 CVW71O 127036953 Ki = 131.83 nM T16691 C7N5DF 127037679 Ki = 324 nM T16691 CTE43C 127037681 Ki = 641 nM T16691 CDAE15 127038033 Ki = 233 nM T16691 CES26L 127039755 Ki = 276 nM T16691 CX1W5M 127040442 Ki = 240 nM T16691 C83YZJ 127045665 Ki = 231 nM T16691 C9EH4D 127045870 Ki = 87 nM T16691 C9CRG7 127045871 Ki = 12 nM T16691 C06KDX 127045872 Ki = 129 nM T16691 CRYE28 127045873 Ki = 54 nM T16691 CX84AD 127045874 Ki = 6 nM T16691 C4Q6DY 127046815 Ki = 290 nM T16691 CF4X5D 127046817 Ki = 7 nM T16691 CZU72I 127046818 Ki > 2000 nM T16691 CF4E8W 127046819 Ki = 5 nM T16691 C38UBC 127046963 Ki = 36 nM T16691 CH6W2T 127046982 Ki = 4 nM T16691 C84PLD 127047536 Ki = 15 nM T16691 C17RWQ 127047537 Ki = 7 nM T16691 C7OCX9 127047538 Ki = 8 nM T16691 CJH46E 127047680 Ki = 3 nM T16691 CUC1G6 127047776 Ki = 16 nM T16691 CV1KL4 127047898 Ki = 11 nM T16691 C3BU0X 127047899 Ki = 48 nM T16691 C7W4MF 127047900 Ki = 24 nM T16691 CLK3C5 127047901 Ki = 2 nM T16691 C5M7AB 129103161 Ki = 241 nM T16691 CI4M9Y 129103313 Ki = 17.7 nM T16691 CR0GI7 129103315 Ki = 29.46 nM T16691 C3WIA6 129103318 Ki = 5.55 nM T16691 C51ZGV 129103322 Ki = 6.36 nM T16691 C50GOC 130442480 Ki = 7900 nM T16691 CM04RF 130442572 Ki = 6900 nM T16691 CCL8F6 132495282 Ki = 39.81 nM T16691 CR7TA8 132495283 Ki = 12.59 nM T16691 C4LJ2Y 132503215 Ki = 401 nM T16691 CM8B1L 132525569 Ki = 121 nM T16691 CU5L0K 132525570 Ki = 12 nM T16691 CAVB41 132584404 Ki > 10000 nM T16691 CS0MB3 132938109 Ki = 295 nM T16691 C5BEG9 134129897 Ki = 8 nM T16691 C6Z5UG 134129927 Ki = 50.12 nM T16691 CPR31M 134130034 Ki = 16 nM T16691 C0QU1J 134130058 Ki = 10 nM T16691 CG4X6D 134130069 Ki = 8 nM T16691 CO3IZ2 134130116 Ki = 10 nM T16691 CM1N3J 134130197 Ki = 8 nM T16691 CZ7GB0 134130237 Ki = 10 nM T16691 CV97TW 134130269 Ki = 13 nM T16691 CL2XT1 134130413 Ki = 6 nM T16691 CJFT74 134130472 Ki = 12 nM T16691 C6XHB4 134130475 Ki = 113 nM T16691 CB2V9D 134130529 Ki = 15 nM T16691 C87WMF 134130564 Ki = 2 nM T16691 CDYJ03 134130753 Ki = 3.8 nM T16691 CP95OK 134130920 Ki = 2 nM T16691 C7NVB0 134131115 Ki = 16 nM T16691 C5Z9WG 134131252 Ki = 2 nM T16691 C4TSE6 134131296 Ki = 39 nM T16691 CA6Z0F 134131307 Ki = 4 nM T16691 CK37GX 134131322 Ki = 11.7 nM T16691 CG5H3O 134131347 Ki = 36 nM T16691 CK57YE 134131472 Ki = 0.5 nM T16691 C2M8RI 134131482 Ki = 36 nM T16691 CLW62U 134131970 Ki = 79.43 nM T16691 C0RQC6 134131976 Ki = 927 nM T16691 C7UOA9 134132432 Ki = 25.12 nM T16691 CTS3J4 134133483 Ki = 1623 nM T16691 CC1DO8 134134456 Ki = 614 nM T16691 C2Q3JY 134135516 Ki = 1633 nM T16691 CJG3U0 134136134 Ki = 1152 nM T16691 CFOU70 134136921 Ki = 3.981 nM T16691 C87ZJW 134137152 Ki = 7.943 nM T16691 C08ZBY 134137332 Ki = 1074 nM T16691 CXF52V 134137560 Ki = 652 nM T16691 CN4LI8 134137732 Ki = 721 nM T16691 C50WSG 134137966 Ki = 1.585 nM T16691 C2DK7E 134139144 Ki = 316.23 nM T16691 CRC2V0 134139826 Ki = 1621 nM T16691 CHK39T 134141166 Ki = 745 nM T16691 C6PSI9 134142907 Ki = 3441 nM T16691 C80TGJ 134144864 Ki = 1706 nM T16691 CK5RU9 134145903 Ki = 480 nM T16691 C2E0ID 134146185 Ki = 2215 nM T16691 CZDH24 134147097 Ki = 1 nM T16691 CV0QZ5 134147124 Ki = 1039 nM T16691 CV4WJ5 134147644 Ki = 316.23 nM T16691 C41XSD 134147935 Ki = 2815 nM T16691 CH21YW 134148634 Ki = 158.49 nM T16691 CBU81N 134149168 Ki > 10000 nM T16691 CSE17M 134150535 Ki = 158.49 nM T16691 C6O8QW 134150900 Ki = 199.53 nM T16691 CE6LN3 134151118 Ki = 1506 nM T16691 C2JN8Y 134151729 Ki = 395 nM T16691 CNC39L 134151926 Ki = 158.49 nM T16691 C76BZW 134151980 Ki = 1724 nM T16691 CIV4H5 134152583 Ki = 2634 nM T16691 C42ZDI 134153624 Ki = 125.89 nM T16691 CX4W7F 134153716 Ki = 843 nM T16691 CM6D4G 134155367 Ki = 10 nM T16691 CIUZ94 134155476 Ki = 561 nM T16691 C90QNV 134155645 Ki = 434 nM T16691 C0AE1P 134156091 Ki = 1 nM T16691 CAB4K6 134156305 Ki = 700 nM T16691 C50XNE 134156520 Ki = 413 nM T16691 CUHE07 134157171 Ki = 640 nM T16691 CL6DN0 134157769 Ki = 1336 nM T16691 C6N8GM 135367405 Ki = 109 nM T16691 C6LU0C 135367816 Ki = 360 nM T16691 CD2TH9 135367820 Ki > 10000 nM T16691 C5AMD9 135367857 Ki = 492 nM T16691 C92ZLY 135437144 Ki = 1.3 nM T16691 C8WL0I 135449090 Ki = 1716 nM T16691 C9ZCL5 135458672 Ki = 3213 nM T16691 CTE23K 135464118 Ki = 742 nM T16691 CF7D9Y 135804742 Ki = 1 nM T16691 CUI8Q2 135847967 Ki = 10 nM T16691 CUKO20 136020617 Ki > 10000 nM T16691 COF0U5 136020618 Ki > 10 nM T16691 CF89JI 136030596 Ki > 10000 nM T16691 CE8GB9 136030693 Ki > 10000 nM T16691 C65VFI 136030744 Ki > 10000 nM T16691 C9G2KR 136046098 Ki = 1.259 nM T16691 COIX80 136054961 Ki > 10000 nM T16691 CS0JL5 136118616 Ki = 1409 nM T16691 CHWC38 136118619 Ki = 2306 nM T16691 CLH0V9 136118648 Ki = 3733 nM T16691 C76XEJ 136118649 Ki = 860 nM T16691 C0W1TM 136118658 Ki = 7523 nM T16691 C42FCS 136118661 Ki = 7300 nM T16691 COX1F8 136118729 Ki = 1405 nM T16691 CN3W5O 136123549 Ki = 1 nM T16691 CB12QP 136152964 Ki = 4476.2 nM T16691 CAE39V 136188797 Ki > 10000 nM T16691 CWP0V5 136216703 Ki > 10000 nM T16691 C7FW4R 136239492 Ki > 10000 nM T16691 CC6OP7 136244089 Ki > 10000 nM T16691 CLAP52 136259032 Ki > 10000 nM T16691 CA18HL 137210067 Ki = 22 nM T16691 CHM36P 137631892 Ki = 791 nM T16691 CD65BY 137632931 Ki = 158 nM T16691 CSL7O5 137633065 Ki = 29.6 nM T16691 CLWC06 137633076 Ki = 1.7 nM T16691 CYNQ85 137633569 Ki = 12 nM T16691 CE61HV 137633644 Ki = 150 nM T16691 CO2X7L 137633663 Ki = 385 nM T16691 CU01TV 137633827 Ki = 4 nM T16691 CQW9J6 137633849 Ki = 91 nM T16691 C6LA9R 137633855 Ki = 239 nM T16691 CFP4L9 137634216 Ki = 326 nM T16691 CYD64J 137634238 Ki = 90.5 nM T16691 C8N4SP 137634321 Ki = 36.1 nM T16691 C9RSC0 137634934 Ki = 29.4 nM T16691 CC51JN 137635185 Ki = 28 nM T16691 C3BOD0 137635355 Ki = 2.5 nM T16691 C94VXJ 137635884 Ki = 60 nM T16691 CYL39G 137635979 Ki = 6 nM T16691 CFM92C 137636384 Ki = 5 nM T16691 CG7T3S 137636699 Ki = 49 nM T16691 CLXP71 137636791 Ki = 17.5 nM T16691 CK6SF0 137637392 Ki = 8.8 nM T16691 C8N1EH 137637698 Ki = 64 nM T16691 CDX39B 137637994 Ki = 3802 nM T16691 CXZ5N7 137638969 Ki = 9.2 nM T16691 C17PBG 137640158 Ki = 20 nM T16691 CEA1L2 137640705 Ki = 305 nM T16691 CKL78U 137640727 Ki = 5 nM T16691 CXP45J 137640850 Ki = 289 nM T16691 C7LN2D 137640966 Ki = 28.2 nM T16691 CYB58F 137641062 Ki = 6.9 nM T16691 C3LYX9 137641832 Ki = 36 nM T16691 C5WS6Q 137642134 Ki = 1863 nM T16691 CCQ2D0 137642224 Ki = 22 nM T16691 CBW26M 137642284 Ki = 100 nM T16691 C35ZUH 137643300 Ki = 18.7 nM T16691 CLPC81 137643504 Ki = 29 nM T16691 CR59HE 137643783 Ki = 30 nM T16691 C7J0MK 137644129 Ki = 96.3 nM T16691 C0VXH9 137644304 Ki = 9.2 nM T16691 CWUM83 137644521 Ki = 20 nM T16691 CUEZ28 137644687 Ki = 133 nM T16691 CDA80E 137644790 Ki = 1041 nM T16691 CZE12U 137645373 Ki = 7.79 nM T16691 CE7G2D 137645440 Ki = 58 nM T16691 CZ8CU6 137645501 Ki = 640 nM T16691 CI4J2N 137645924 Ki = 30 nM T16691 CCP38D 137645926 Ki = 1020 nM T16691 CGC4W8 137645927 Ki = 1.3 nM T16691 CVX74E 137646045 Ki = 1 nM T16691 CLT73G 137647199 Ki = 2 nM T16691 CUDM82 137647787 Ki = 11.6 nM T16691 CVOX24 137648172 Ki = 5.7 nM T16691 CP7U1T 137648205 Ki = 277 nM T16691 CJ83AX 137648352 Ki = 398 nM T16691 CN19AD 137648438 Ki = 37.8 nM T16691 CQU92A 137649408 Ki = 11.5 nM T16691 CJCU15 137649536 Ki = 56 nM T16691 CMXI62 137649997 Ki = 6712 nM T16691 CM4YW3 137650127 Ki = 119 nM T16691 C3JKC5 137650191 Ki = 52 nM T16691 C52IRM 137650705 Ki = 445 nM T16691 CP2WU7 137650747 Ki = 4.5 nM T16691 CE0UW8 137650795 Ki = 35.7 nM T16691 CTSB07 137650870 Ki = 348 nM T16691 CKG08R 137650961 Ki = 8279 nM T16691 C24NHR 137651282 Ki = 88 nM T16691 CH96PE 137651330 Ki = 64 nM T16691 CZM2Q5 137651613 Ki = 6.7 nM T16691 CU4S1W 137651887 Ki = 36 nM T16691 CVK26R 137652044 Ki = 2412 nM T16691 CHFK13 137652210 Ki = 266 nM T16691 CZLK69 137652249 Ki = 18.4 nM T16691 C51CGJ 137652310 Ki = 1459 nM T16691 CAE1F8 137652414 Ki = 50 nM T16691 CZ5K3F 137653132 Ki = 55.6 nM T16691 CA7JP5 137653219 Ki = 7.8 nM T16691 C2E3FV 137653850 Ki = 1185 nM T16691 COLJ56 137654026 Ki = 95 nM T16691 CKN9V4 137654042 Ki = 100 nM T16691 CX82HS 137654666 Ki = 250 nM T16691 C0SKV1 137654850 Ki = 52 nM T16691 CX5YF2 137655402 Ki = 4 nM T16691 C4VG0U 137655411 Ki = 309 nM T16691 C48TXI 137655693 Ki = 1828 nM T16691 CK5L7D 137655929 Ki = 440 nM T16691 CV4XE1 137656063 Ki = 16.3 nM T16691 C5D2GX 137656602 Ki = 59.7 nM T16691 CQ3HV5 137656608 Ki = 7.8 nM T16691 CIW45A 137656837 Ki = 5.7 nM T16691 CO3L7F 137656918 Ki = 755 nM T16691 C1UZX3 137657317 Ki = 312 nM T16691 C5V6CH 137657598 Ki = 32 nM T16691 CG07QC 137657740 Ki = 193 nM T16691 CFC57K 137658350 Ki = 194 nM T16691 C72MIH 137658424 Ki = 28 nM T16691 CKVH89 137658916 Ki = 2 nM T16691 C4JO1X 137659244 Ki = 80 nM T16691 C4JVW5 137659459 Ki = 64 nM T16691 CL6Y2M 137659696 Ki = 34.9 nM T16691 CB4HN7 137660291 Ki = 19 nM T16691 CX4D7Y 137660741 Ki = 1016 nM T16691 CA4MT5 137661210 Ki = 1.63 nM T16691 CC1X5S 137661237 Ki = 14.3 nM T16691 CO9R5P 137661730 Ki = 348 nM T16691 C78CZR 137661837 Ki = 31.2 nM T16691 CNA2D1 137662033 Ki = 64 nM T16691 C8ZIY5 137662324 Ki = 365 nM T16691 C0R6XM 138691314 Ki = 1660 nM T16691 CU3Y7W 138691316 Ki = 1349 nM T16691 CH2W4P 138691317 Ki = 3020 nM T16691 CHSC40 138691321 Ki = 2455 nM T16691 C18UZA 138691329 Ki = 4169 nM T16691 C1XWV0 138691338 Ki = 6918 nM T16691 C6LE1A 138691362 Ki > 10000 nM T16691 CN9R4A 138691364 Ki = 7762 nM T16691 C8H2KR 138691366 Ki = 4898 nM T16691 C2Z9CD 139488518 Ki = 6457 nM T16691 CJK95T 139488527 Ki > 10000 nM T16691 CZ6H9M 139488539 Ki = 2951 nM T16691 CAF2H8 139488606 Ki = 2884 nM T16691 C54CIL 139488740 Ki > 10000 nM T16691 CK42UE 142592111 Ki = 2.6 nM T16691 CM03WS 142592130 Ki = 1.9 nM T16691 CL8Y2Z 145949620 Ki = 80 nM T16691 C6IFL5 145950947 Ki = 26 nM T16691 CSA0M6 145951217 Ki = 126 nM T16691 CD69JU 145951815 Ki = 1298 nM T16691 CTPH52 145952652 Ki = 139 nM T16691 CG36FD 145953693 Ki = 62 nM T16691 CF67VS 145953749 Ki = 36 nM T16691 CA2J5S 145954503 Ki = 9000 nM T16691 CRQ16N 145954675 Ki = 0.2 nM T16691 CY71FH 145955674 Ki = 320 nM T16691 C8ZXQ4 145955822 Ki = 33 nM T16691 C6A4BR 145957184 Ki = 42 nM T16691 CGU2Y4 145958161 Ki = 30 nM T16691 C5CH7K 145958329 Ki = 80 nM T16691 C2YCL8 145959790 Ki = 312 nM T16691 C9X7KL 145959871 Ki = 110 nM T16691 CQ9P6R 145960299 Ki = 1251 nM T16691 CBX8F6 145960391 Ki = 49 nM T16691 C67GQI 145961372 Ki = 1837 nM T16691 CEYW94 145961507 Ki = 137 nM T16691 CNVZ94 145961959 Ki = 61 nM T16691 C8BWY4 145962006 Ki = 427 nM T16691 C6QCV1 145962275 Ki = 269 nM T16691 CC75OQ 145962993 Ki = 365 nM T16691 CD45OW 145963033 Ki = 131 nM T16691 C5LJY2 145963274 Ki = 45 nM T16691 CW3K5O 145963649 Ki = 711 nM T16691 C7KC3T 145963830 Ki = 2200 nM T16691 C4Y2AL 145964000 Ki > 5000 nM T16691 CHDN35 145964150 Ki > 10000 nM T16691 C1KH2E 145964159 Ki = 2600 nM T16691 C95NZO 145964427 Ki = 1540 nM T16691 C6T4RY 145964846 Ki > 5000 nM T16691 C12OVL 145965034 Ki > 10000 nM T16691 C9D8IB 145965203 Ki > 5000 nM T16691 CA8KF0 145965309 Ki > 5000 nM T16691 CLP94W 145965668 Ki = 2843 nM T16691 C8TF9G 145965840 Ki = 1693 nM T16691 C5W4LM 145965940 Ki > 10000 nM T16691 C1T4DN 145966418 Ki = 2005 nM T16691 C81VUO 145967771 Ki > 10 nM T16691 CJS56K 145967795 Ki > 10000 nM T16691 CQ8EM6 145969402 Ki = 4737 nM T16691 C1T7GL 145971527 Ki = 1800 nM T16691 C8A2XG 145971561 Ki = 1131 nM T16691 CQJ5O8 145971635 Ki > 10000 nM T16691 CUZ2E9 145971739 Ki = 374 nM T16691 C56RAO 145972025 Ki = 4577 nM T16691 C79TNE 145972796 Ki > 10000 nM T16691 CB3KH0 145973178 Ki = 5 nM T16691 CEOY46 145973577 Ki = 200 nM T16691 CT5CX0 145973771 Ki = 7900 nM T16691 C6XIN0 145974114 Ki > 10000 nM T16691 CW6EX3 145974189 Ki = 268 nM T16691 CD8ZL6 145974750 Ki > 10 nM T16691 C6ZEI2 145974789 Ki = 317 nM T16691 C6PH4F 145975226 Ki > 10000 nM T16691 COY2P3 145975720 Ki = 4744 nM T16691 CL7EX5 145975776 Ki = 2155 nM T16691 C7R2MD 145975905 Ki = 6556 nM T16691 C71CYU 145975946 Ki > 10000 nM T16691 C0V4AL 145975992 Ki = 5285 nM T16691 C2TN8W 145976085 Ki > 10000 nM T16691 C8XFM7 145976120 Ki > 5000 nM T16691 CZ5XK2 145976408 Ki = 5559 nM T16691 C34XME 145976696 Ki = 2427 nM T16691 CXDR94 145977222 Ki > 5000 nM T16691 C8NW7Y 145977256 Ki = 6267 nM T16691 C6BFY7 145977338 Ki > 10000 nM T16691 C0Y6QO 145977799 Ki > 10000 nM T16691 C3BI1R 145978113 Ki > 10000 nM T16691 C8VL3Y 145978472 Ki = 7746 nM T16691 CQU8R0 145978665 Ki > 10000 nM T16691 C6AV9G 145978819 Ki > 10000 nM T16691 C87MSW 145980271 Ki = 1670 nM T16691 CEK60A 145982506 Ki = 2310 nM T16691 CI59TX 145983018 Ki = 3912 nM T16691 CYC58R 145983059 Ki = 130 nM T16691 C4F5OT 145983128 Ki = 641 nM T16691 C5ZG9M 145983139 Ki = 291 nM T16691 CV2GU9 145983144 Ki = 77 nM T16691 C4PKM2 145983390 Ki = 623 nM T16691 CIAF74 145983468 Ki = 344 nM T16691 CE7MF4 145983751 Ki = 1259 nM T16691 CDQ4U7 145983760 Ki = 176 nM T16691 CYW9B2 145983794 Ki = 221 nM T16691 C8I1WG 145983961 Ki = 40 nM T16691 CP5H4D 145984065 Ki = 23 nM T16691 CJ35DM 145984299 Ki = 313 nM T16691 CU7E4M 145984511 Ki = 348 nM T16691 C6JUY0 145984737 Ki = 360 nM T16691 CID02G 145984807 Ki = 2990 nM T16691 CM5X3V 145985050 Ki = 137 nM T16691 CG10LK 145985224 Ki = 457 nM T16691 CFJ9B3 145985233 Ki = 169 nM T16691 C5AOI6 145985289 Ki = 190 nM T16691 CW30NA 145985505 Ki = 92 nM T16691 C7ZRP1 145985527 Ki = 18 nM T16691 C2XY8Q 145985533 Ki = 311 nM T16691 C7NI4X 145985585 Ki = 497 nM T16691 C9LJ5T 145985692 Ki = 40 nM T16691 C7QIX0 145985718 Ki = 949 nM T16691 C6V5QS 145985823 Ki = 45 nM T16691 C07GKD 145985958 Ki = 1810 nM T16691 CCM18E 145986031 Ki = 337 nM T16691 CR0XQ3 145986138 Ki = 104 nM T16691 CNJH37 145986752 Ki = 1400 nM T16691 CUGO10 145988693 Ki = 1680 nM T16691 C4GV8Q 145990586 Ki = 862 nM T16691 CC2G1V 146025727 Ki = 7200 nM T16691 C5ZOJ3 146680920 Ki = 3 nM T16691 CD1CB9 151199471 Ki = 20 nM T16691 C6P3SR 153287553 Ki > 10000 nM T16691 CV9G7Z 153287572 Ki > 10000 nM T16691 CO85KL 153287574 Ki > 10000 nM T16691 CZ1K4D 155510674 Ki = 1716 nM T16691 CC3KP7 155510927 Ki = 2 nM T16691 CM4RB0 155511262 Ki = 55 nM T16691 CNE0U3 155511424 Ki = 109 nM T16691 C9KX6O 155511928 Ki = 433 nM T16691 CXF90M 155512487 Ki = 2 nM T16691 CO68LC 155512944 Ki = 550 nM T16691 CP0W8C 155513247 Ki = 132 nM T16691 C90FST 155513438 Ki = 5 nM T16691 C95QOT 155514378 Ki = 4 nM T16691 C3SQI7 155514459 Ki = 14 nM T16691 C0F8BR 155514505 Ki = 1032 nM T16691 CI4DT8 155514575 Ki = 10 nM T16691 CJUI87 155514774 Ki = 58 nM T16691 CQ9ZH8 155514839 Ki = 18 nM T16691 C4X2RG 155515318 Ki = 60 nM T16691 C3NB0D 155515324 Ki = 3574 nM T16691 CZQ32K 155515399 Ki = 475 nM T16691 C0Q8PR 155515407 Ki = 3187 nM T16691 CWO56B 155515415 Ki = 250 nM T16691 C2TN5D 155515890 Ki = 1461 nM T16691 C7KT0D 155515919 Ki = 10 nM T16691 C13LOV 155515942 Ki = 20 nM T16691 C7OF4C 155516118 Ki = 25 nM T16691 CG5M1O 155516282 Ki = 3666 nM T16691 CCS1D6 155517413 Ki = 20 nM T16691 CW0B5K 155518159 Ki = 25 nM T16691 CY7PH5 155518290 Ki = 24 nM T16691 CYB12O 155518974 Ki = 5765 nM T16691 C2E6UC 155519088 Ki = 18 nM T16691 CCEZ93 155519102 Ki = 23 nM T16691 CQD2J7 155519393 Ki = 101 nM T16691 C2SXT1 155519515 Ki = 374 nM T16691 C0KLD8 155519559 Ki = 2 nM T16691 C07BTO 155519598 Ki = 2214 nM T16691 CUSA24 155519891 Ki > 10000 nM T16691 C5FL7R 155520499 Ki = 494 nM T16691 C8OC3W 155520552 Ki = 237 nM T16691 CQ76MP 155521503 Ki = 9 nM T16691 C1OS6D 155522116 Ki = 34 nM T16691 C98RDQ 155522218 Ki = 435 nM T16691 CHA82N 155522233 Ki = 1696 nM T16691 C2TV4Y 155522487 Ki = 50 nM T16691 CK26JU 155522511 Ki = 693 nM T16691 CP6H1D 155522562 Ki = 624 nM T16691 CUG8L3 155522920 Ki = 23 nM T16691 CUG4Q8 155523121 Ki = 21 nM T16691 CN4Y6C 155523355 Ki = 11 nM T16691 CD9QU6 155523519 Ki = 157 nM T16691 C76ARL 155523771 Ki = 220 nM T16691 C5KYB4 155524228 Ki = 71 nM T16691 CK4B0R 155524491 Ki = 1030 nM T16691 CUO93F 155524808 Ki = 921 nM T16691 CQB0M8 155524884 Ki = 78 nM T16691 C65UZD 155524956 Ki = 507 nM T16691 C7FAU5 155525318 Ki = 6 nM T16691 CG2ZS4 155525596 Ki = 522 nM T16691 CZ81JA 155526026 Ki = 459 nM T16691 CN6Z4X 155526468 Ki = 44 nM T16691 C1U2XO 155526651 Ki = 999 nM T16691 CS1GY7 155527191 Ki = 199 nM T16691 CI4UY3 155527359 Ki = 145 nM T16691 C10BPO 155527391 Ki = 37 nM T16691 CW68KC 155528355 Ki = 10 nM T16691 CF29DP 155528725 Ki = 152 nM T16691 C7C1EF 155528967 Ki = 697 nM T16691 C5J7AU 155529153 Ki = 111 nM T16691 C9KS5C 155529450 Ki = 52 nM T16691 CKZ25Y 155529679 Ki = 1272 nM T16691 C7UZI1 155530285 Ki = 157 nM T16691 C3X4IA 155530328 Ki = 372 nM T16691 C9PC3D 155530350 Ki = 937 nM T16691 C57ETL 155530553 Ki = 303 nM T16691 CVLC03 155530779 Ki = 76 nM T16691 C98YQF 155531012 Ki = 132 nM T16691 C4W6VC 155531065 Ki = 7 nM T16691 C5HWP4 155531362 Ki = 9 nM T16691 CQ86CH 155531455 Ki = 16 nM T16691 CCT8V9 155531846 Ki = 507 nM T16691 C5XNT1 155532396 Ki = 105 nM T16691 CS86HA 155532544 Ki = 345 nM T16691 CX35QS 155532545 Ki = 79 nM T16691 CFI23P 155532887 Ki = 556 nM T16691 C3W6HV 155532983 Ki = 100 nM T16691 CX6DV4 155533028 Ki = 952 nM T16691 C23GDV 155533534 Ki = 1651 nM T16691 CSY06A 155533573 Ki = 15 nM T16691 C3OEH2 155533648 Ki = 1410 nM T16691 C15RYP 155533660 Ki = 10 nM T16691 CX1U4H 155533704 Ki = 596 nM T16691 CY01GZ 155533850 Ki = 1320 nM T16691 C2GIL4 155533990 Ki = 247 nM T16691 C6ACO9 155534040 Ki = 65 nM T16691 CP3J8B 155534152 Ki = 29 nM T16691 C3L0CP 155534184 Ki = 1030 nM T16691 C9BGE1 155534201 Ki = 30 nM T16691 CG85SB 155534301 Ki = 5253 nM T16691 C3VGT0 155534362 Ki = 1709 nM T16691 CW7SV9 155534575 Ki = 104 nM T16691 C5HS8N 155534670 Ki = 5 nM T16691 C75FSY 155534794 Ki = 8 nM T16691 C6KF4E 155535154 Ki = 452 nM T16691 C14JEX 155535878 Ki = 4 nM T16691 CB79ZW 155536080 Ki > 10000 nM T16691 C5I1JA 155536087 Ki = 1619 nM T16691 C72FLG 155536152 Ki = 128 nM T16691 C7FVE8 155537034 Ki = 6910 nM T16691 C36FRH 155537074 Ki = 14 nM T16691 CD75GP 155537227 Ki = 15 nM T16691 CB8IC7 155538144 Ki = 3467 nM T16691 C5F2GI 155538236 Ki = 1146 nM T16691 C9TIU2 155538367 Ki = 1622 nM T16691 CYC1P3 155538451 Ki = 246 nM T16691 CM08NT 155538716 Ki = 280 nM T16691 CQ69UA 155538814 Ki = 148 nM T16691 C0D6AQ 155538873 Ki = 10 nM T16691 CAT98F 155539483 Ki = 301 nM T16691 CC1VR4 155539573 Ki = 201 nM T16691 C6S8BA 155539600 Ki = 19 nM T16691 C2HE6C 155540062 Ki = 7 nM T16691 C42GUK 155540147 Ki = 603 nM T16691 CJD9C8 155540541 Ki = 186 nM T16691 CCFM15 155540673 Ki = 21 nM T16691 C2OWD4 155540721 Ki = 17 nM T16691 CR2K1T 155540795 Ki = 19 nM T16691 CNU92V 155540807 Ki = 81 nM T16691 COS2E7 155541072 Ki = 7271 nM T16691 CMP8Q2 155541547 Ki = 83 nM T16691 C6SU1V 155541676 Ki = 501 nM T16691 CP7UG2 155541866 Ki = 90 nM T16691 COZ46W 155541871 Ki = 480 nM T16691 C58YSH 155542160 Ki = 4.8 nM T16691 CB62ZS 155542237 Ki = 21 nM T16691 CX61OI 155542267 Ki = 219 nM T16691 CXCW81 155542321 Ki = 11 nM T16691 C9FS3Y 155542461 Ki = 14 nM T16691 CGC1P6 155543054 Ki = 334 nM T16691 CUI2G9 155543192 Ki = 556 nM T16691 CDO05U 155543223 Ki = 266 nM T16691 CT6HY4 155543250 Ki = 245 nM T16691 C68MSK 155543653 Ki = 118 nM T16691 CIEQ43 155543869 Ki = 31 nM T16691 CZ7O0A 155544139 Ki = 355 nM T16691 CD84VK 155544810 Ki = 1681 nM T16691 CP54KO 155544836 Ki = 102 nM T16691 C2XZD8 155545087 Ki = 225 nM T16691 CO9X1Z 155545526 Ki = 263 nM T16691 CI0YL8 155545625 Ki = 7079 nM T16691 CFQE48 155545832 Ki = 13 nM T16691 C86MKF 155546176 Ki = 175 nM T16691 C74GFO 155546189 Ki = 710 nM T16691 CJBP49 155546194 Ki = 128 nM T16691 CH3W9N 155546350 Ki > 10000 nM T16691 C1SVX6 155547259 Ki = 8.2 nM T16691 CD02EN 155547436 Ki = 347 nM T16691 COJ27N 155547693 Ki = 207 nM T16691 CM4XB6 155548127 Ki = 4.6 nM T16691 CJ7AL8 155548205 Ki = 71 nM T16691 CAT9X4 155548275 Ki = 107 nM T16691 C5LYE8 155548677 Ki = 21 nM T16691 C87JGN 155549153 Ki = 585 nM T16691 CGP8O5 155549315 Ki = 3270 nM T16691 C52FRY 155549978 Ki = 971 nM T16691 CU93YK 155550351 Ki = 12 nM T16691 CY34NR 155550580 Ki = 28 nM T16691 CHXB35 155551102 Ki = 21 nM T16691 C8HPN7 155551113 Ki = 1726 nM T16691 CYOW72 155551197 Ki = 418 nM T16691 CUZJ87 155551219 Ki = 12 nM T16691 C61IVC 155551353 Ki = 407 nM T16691 CHS71N 155551685 Ki = 920 nM T16691 CMCG80 155551834 Ki = 22 nM T16691 C6E9LK 155552054 Ki = 1699 nM T16691 CA1WS9 155552212 Ki = 918 nM T16691 CY94BV 155552356 Ki = 440 nM T16691 CMS62Z 155552380 Ki = 23 nM T16691 CF40VB 155552641 Ki = 69 nM T16691 CDQ7C2 155552798 Ki = 2045 nM T16691 CPV35U 155552826 Ki = 6062 nM T16691 CT23YW 155553005 Ki = 1463 nM T16691 C6STK4 155553745 Ki = 1034 nM T16691 C48LRX 155554020 Ki = 289 nM T16691 CDV6B9 155554036 Ki = 129 nM T16691 CL3FC8 155554246 Ki = 264 nM T16691 CKF75H 155554324 Ki = 689 nM T16691 C6ZSU3 155554462 Ki = 26 nM T16691 C0P6IW 155554556 Ki = 240 nM T16691 CCA21K 155554569 Ki = 2.3 nM T16691 CRY82F 155554955 Ki = 42 nM T16691 CC70RV 155555136 Ki = 8 nM T16691 CLN79H 155555200 Ki = 527 nM T16691 C1RCM0 155555224 Ki = 60 nM T16691 CWL03Q 155555238 Ki = 9 nM T16691 C5Q4UP 155555402 Ki = 2.7 nM T16691 C2E5TR 155555506 Ki = 61 nM T16691 CUNK28 155555525 Ki = 9 nM T16691 CF6R7E 155556168 Ki = 58 nM T16691 CO52HW 155556527 Ki = 794 nM T16691 C1N5VF 155556756 Ki = 50 nM T16691 C2GE4Q 155557005 Ki = 0.43 nM T16691 C5QYS0 155557134 Ki = 476 nM T16691 C59EUZ 155557143 Ki = 210 nM T16691 CD2L3K 155557443 Ki = 3802 nM T16691 CER48T 155557500 Ki = 455 nM T16691 C64EMC 155557523 Ki = 82 nM T16691 CJ0LE3 155557661 Ki = 419 nM T16691 C6END5 155557760 Ki = 7 nM T16691 CHC8S1 155557772 Ki = 11 nM T16691 CF08HV 155557890 Ki = 531 nM T16691 CJZ12T 155558380 Ki = 254 nM T16691 CF6H3V 155558408 Ki = 911 nM T16691 C06BZW 155559811 Ki = 129 nM T16691 CFU9P0 155560188 Ki = 14 nM T16691 C1Z2GD 155560272 Ki = 594 nM T16691 CL4I0D 155560922 Ki = 13 nM T16691 COG70U 155560942 Ki = 3 nM T16691 C2HF6P 155561581 Ki = 242 nM T16691 C5O8AU 155561865 Ki = 759 nM T16691 COL7N8 155561901 Ki = 3467 nM T16691 CXPT57 155561906 Ki = 112 nM T16691 CL45NV 155561914 Ki = 1128 nM T16691 CW7M1D 155561995 Ki = 728 nM T16691 CRTD49 155562063 Ki = 486 nM T16691 C93KWN 155562202 Ki = 671 nM T16691 CO3C6L 155562423 Ki = 31 nM T16691 C5AI0S 155562519 Ki = 85 nM T16691 C4ZA0Q 155562620 Ki = 13 nM T16691 C5BQ8U 155562652 Ki = 690 nM T16691 C5E6BI 155562755 Ki = 45 nM T16691 CF6B4W 155562834 Ki = 182 nM T16691 CZ6IA2 155562918 Ki = 87 nM T16691 CRCW25 155562997 Ki = 29 nM T16691 CBH14K 155563164 Ki = 83 nM T16691 CG1L8E 155563286 Ki = 5888 nM T16691 C38WXS 155563374 Ki = 9 nM T16691 C0INS4 155563826 Ki = 93 nM T16691 C2QLX9 155565138 Ki = 25 nM T16691 CIB3R0 155565292 Ki = 74 nM T16691 C2MIU5 155565813 Ki = 2 nM T16691 C7P5VG 155566191 Ki = 3 nM T16691 C7O6YP 155566439 Ki = 235 nM T16691 CU46EB 155566665 Ki = 3 nM T16691 CEV3B9 155566852 Ki = 25 nM T16691 C67LAG 155566854 Ki = 14 nM T16691 CW1TN7 155566925 Ki = 794 nM T16691 C41UWT 155567307 Ki = 1916 nM T16691 C6I5QA 155567666 Ki = 170 nM T16691 CW3Q7C 155567905 Ki = 18 nM T16691 CA68TK 155568224 Ki = 126 nM T16691 C4EX7C 155568246 Ki = 427 nM T16691 C6V5KP 155568249 Ki = 247 nM T16691 CP03VZ 155568299 Ki = 9 nM T16691 CVU42Z 155568628 Ki = 125 nM T16691 CXP3E4 155568794 Ki = 121 nM T16691 CB5IP9 155569021 Ki = 1860 nM T16691 C0CZK6 155569337 Ki = 18 nM T16691 CP9V7M 155569396 Ki = 1380 nM T16691 C3ZNX6 155569414 Ki = 2352 nM T16691 CZ8RV4 155569568 Ki = 67 nM T16691 C3N9VU 10251906 Ki = 73 nM T16691 CP9TR0 10324985 Ki = 120.3 nM T16691 D00AVR 135476741 Ki = 8768 nM T16691 D00CRA 1574 Ki = 46 nM T16691 D00DZY 11849201 Ki = 4000 nM T16691 D00GSD 25107716 Ki = 1571 nM T16691 D00OBS 44559159 Ki > 10000 nM T16691 D00OCC 9948345 Ki = 1.2 nM T16691 D00VRV 10171 Ki = 17 nM T16691 D01DCE 44401620 Ki = 4200 nM T16691 D01KAX 135453290 Ki > 10000 nM T16691 D01KVG 9843179 Ki = 524.81 nM T16691 D01TYJ 44405257 Ki = 980 nM T16691 D01WWC 16573 Ki = 306 nM T16691 D01ZMO 44401549 Ki = 11800 nM T16691 D02JFD 6918649 Ki = 0.7 nM T16691 D02SBM 49836719 Ki = 27 nM T16691 D02UWB 1809 Ki = 720 nM T16691 D02VHJ 21071574 Ki = 10 nM T16691 D02YSX 197033 Ki = 26 nM T16691 D03DET 10287730 Ki < 10000 nM T16691 D03LPH 107838 Ki > 5000 nM T16691 D03TDN 1342 Ki = 100 nM T16691 D03TSY 24825775 Ki > 1000 nM T16691 D04AQE 1833 Ki < 50 nM T16691 D05DAF 11849198 Ki = 2840 nM T16691 D05EQG 5265 Ki = 1595 nM T16691 D05GDP 599482 Ki > 10000 nM T16691 D05HJP 6476992 Ki = 640 nM T16691 D05JPG 44401277 Ki = 3 nM T16691 D05SAP 11849791 Ki = 290 nM T16691 D05XGR 6918647 Ki = 5 nM T16691 D06FXO 10042892 Ki = 13 nM T16691 D06QVB 44390054 Ki = 34 nM T16691 D06VDN 443391 IC50 = 667 nM T16691 D07DCN 11849196 Ki = 62 nM T16691 D07LIE 11849199 Ki = 50 nM T16691 D07LRJ 5312149 Ki = 0.631 nM T16691 D08BCF 5011 Ki = 3600 nM T16691 D08OFG 11177588 Ki > 10000 nM T16691 D08SMK 14571158 Ki = 8 nM T16691 D08VGJ 9904281 Ki = 1157 nM T16691 D09HJL 10331436 Ki = 2200 nM T16691 D09LVG 44401550 Ki = 4470 nM T16691 D09RPR 16737207 Ki > 10000 nM T16691 D09RXU 45488131 Ki = 31 nM T16691 D09VSK 4301799 Ki = 2530 nM T16691 D09WIL 10028436 Ki = 851.14 nM T16691 D0B1KT 15953802 Ki = 100000000 nM T16691 D0C4AE 10246639 Ki = 91 nM T16691 D0C5GF 6918515 Ki = 20 nM T16691 D0C5XQ 1832 Ki = 13 nM T16691 D0C8UV 5113605 Ki = 6.9 nM T16691 D0CK9K 6918513 Ki = 16 nM T16691 D0CY6E 44414681 Ki = 37 nM T16691 D0D2XH 44413494 Ki = 3.3 nM T16691 D0D3YN 1238 Ki < 50 nM T16691 D0D6FC 15281645 Ki = 38 nM T16691 D0E0DR 11849194 Ki = 21 nM T16691 D0F0IA 11301655 Ki > 2000 nM T16691 D0F1FN 15893127 Ki > 5000 nM T16691 D0F6CD 5202 Ki = 33 nM T16691 D0F6GP 49836621 Ki = 4.9 nM T16691 D0FF6S 16038374 IC50 > 10000 nM T16691 D0FV7K 19779451 Ki = 8200 nM T16691 D0G6NV 44413495 Ki = 1.8 nM T16691 D0G7QT 10131112 IC50 = 7.4 nM T16691 D0H0IZ 11849794 Ki = 70 nM T16691 D0H3WJ 44435193 Ki = 1200 nM T16691 D0H5EP 44388931 Ki = 12 nM T16691 D0H7PC 6918553 Ki = 2.6 nM T16691 D0H9QG 5312148 Ki < 15848.93 nM T16691 D0I9IF 56655571 Ki = 0.2089 nM T16691 D0J6JT 1355 Ki = 2300 nM T16691 D0J7EM 24776941 Ki = 90 nM T16691 D0J9MP 11849197 Ki = 230 nM T16691 D0JT3M 20722800 Ki = 32 nM T16691 D0K5NZ 68848 Ki = 776 nM T16691 D0KS0I 24894910 EC50 > 10000 nM T16691 D0L5MW 181743 Ki = 257 nM T16691 D0L7PA 3248571 Ki = 2.512 nM T16691 D0LA4I 44401621 Ki = 740 nM T16691 D0N7NK 10202564 EC50 = 0.06457 nM T16691 D0N8AO 11849789 Ki = 85 nM T16691 D0O3GF 1220 Ki > 10000 nM T16691 D0O3GQ 11849796 Ki = 115 nM T16691 D0OG0R 10337743 Ki = 4.8 nM T16691 D0P8JA 5312145 IC50 = 26.3 nM T16691 D0PQ1U 11818252 Ki = 3 nM T16691 D0Q7AF 6918836 Ki = 0.2 nM T16691 D0R3GW 10296414 Ki < 10000 nM T16691 D0R7VT 44263491 Ki = 10 nM T16691 D0S4XR 25263303 Ki = 1.3 nM T16691 D0SJ6E 44438719 Ki = 2.5 nM T16691 D0T7VZ 44397102 Ki = 6 nM T16691 D0TG0I 10154392 Ki = 0.3 nM T16691 D0TX8W 594590 Ki = 2700 nM T16691 D0V2PB 5312144 Ki = 12 nM T16691 D0V4RP 1346 Ki = 1.2 nM T16691 D0V5AN 44567986 Ki = 29 nM T16691 D0VI0S 49836506 Ki = 134 nM T16691 D0W2HW 6090 Ki = 575 nM T16691 D0W2QN 44403334 IC50 = 300 nM T16691 D0X1IU 44401390 Ki = 6100 nM T16691 D0X6MT 4106 Ki = 0.4 nM T16691 D0XJ6D 10356663 Ki = 12 nM T16691 D0Y1LJ 10017687 Ki = 25 nM T16691 D0Y4WH 9840311 Ki = 5 nM T16691 D0Y9TL 13702393 Ki > 10000 nM T16691 D0ZC9Q 44393574 Ki = 1900 nM T39921 D0A9KI 9863367 IC50 = 160 nM T39921 D0T3ME 156422 IC50 = 58 nM T39921 C61KPI 24856363 IC50 = 53 nM T39921 CH1YI6 24856364 IC50 = 27 nM T39921 C9VXN3 44578709 IC50 = 6 nM T39921 CDC2V8 44593640 IC50 = 88 nM T39921 C69HNG 56967399 IC50 = 200 nM T62974 D02XIY 448601 Ki = 66 nM T62974 D0TV0C 9941444 Ki < 100 nM T62974 D06JFI 11251755 IC50 = 1.8 nM T62974 D0J8PI 158782 IC50 > 1000 nM T62974 D09JXL 5311430 Ki < 1000 nM T62974 D0Y2HR 2247 Ki > 10000 nM T62974 C6XYL5 6918011 Ki < 1000 nM T62974 CHM63P 6918026 Ki = 158.49 nM T62974 CR0U6E 9827283 Ki = 6840 nM T62974 CA8UQ7 9848232 Ki > 10000 nM T62974 CTRI07 9852911 Ki = 1100 nM T62974 C9BJ3Q 9854636 IC50 = 0.84 nM T62974 CS2D0V 9872511 Ki = 118 nM T62974 C71BKL 9893924 Ki = 6 nM T62974 CMLP16 9918828 Ki < 100 nM T62974 CRP01W 9959684 Ki = 413 nM T62974 C3Z5YJ 9963342 Ki = 501.19 nM T62974 CIT57N 9985523 Ki = 1700 nM T62974 C64LIB 10009650 Ki = 100 nM T62974 C58EOI 10053855 Ki = 1400 nM T62974 CL6G0Z 10094509 Ki = 5010 nM T62974 C9C7RK 10096510 Ki > 10000 nM T62974 CFZN71 10166743 Ki = 3840 nM T62974 CI21CK 10179247 Ki > 10000 nM T62974 C6DRE9 10210016 Ki > 10000 nM T62974 C4M9GN 10248767 Ki > 10000 nM T62974 CSY5K2 10325243 Ki = 2000 nM T62974 C67NLY 10369961 Ki = 16 nM T62974 CL87OB 10411795 Ki > 10000 nM T62974 CP2S9D 10436888 Ki = 14 nM T62974 C0YFD4 10505242 Ki = 4200 nM T62974 CN3IV5 10528970 Ki = 7000 nM T62974 CJ40IE 10531093 Ki = 53 nM T62974 CS96ON 10534086 IC50 = 1000 nM T62974 CRZ9I3 10553122 Ki = 4000 nM T62974 CB2NK4 10554498 Ki = 70 nM T62974 CA1VI4 10554709 Ki = 1000 nM T62974 CHZ9I8 10554930 Ki = 3000 nM T62974 CY3ZE9 10577746 IC50 = 1047 nM T62974 CIY02U 10578474 Ki = 477 nM T62974 C9C0HF 10580397 Ki = 500 nM T62974 CUW4E5 10601454 Ki = 2000 nM T62974 CD8ZW7 10602230 Ki = 476 nM T62974 CVY6D0 10603005 Ki = 1200 nM T62974 CGZ6W8 10625454 Ki = 176 nM T62974 C0SXF1 10625762 Ki = 1000 nM T62974 CU3DQ6 10630127 Ki = 1000 nM T62974 C15AHJ 10650427 Ki = 1700 nM T62974 C7AX8J 10650940 Ki = 132 nM T62974 C5UOS4 10698494 Ki = 185 nM T62974 CT81RB 10698706 Ki = 15000 nM T62974 C45JIZ 10699714 Ki = 2000 nM T62974 CG2UX4 10701257 IC50 = 1000 nM T62974 C27FVZ 10720221 Ki = 7000 nM T62974 CP0F7C 10724811 IC50 = 1000 nM T62974 C3TMY5 10724880 IC50 = 1000 nM T62974 CK7R2B 10745635 Ki = 1400 nM T62974 CJM47E 10748701 IC50 = 1000 nM T62974 CWF2N5 10748831 IC50 = 943 nM T62974 CLQ07H 10768264 Ki = 803 nM T62974 C4X2CO 10769191 Ki = 514 nM T62974 CLW4V6 10770814 Ki = 1900 nM T62974 CO56HI 10772403 IC50 = 1000 nM T62974 CGN0Z5 10772578 IC50 = 1000 nM T62974 COY17C 10793795 Ki = 71000 nM T62974 C3L4DH 10796238 IC50 = 1000 nM T62974 C0WND2 10815650 Ki = 113 nM T62974 C61EOJ 10816544 Ki = 1700 nM T62974 C15QGO 10819673 IC50 = 1000 nM T62974 CJ4T3I 10841338 Ki = 520 nM T62974 CFL71O 10843862 IC50 = 1000 nM T62974 CRP17A 10865371 Ki = 1260 nM T62974 CDE2S9 10876118 Ki = 1040 nM T62974 C2PJ1O 10876898 Ki = 630.96 nM T62974 CEV12M 10887003 Ki = 680 nM T62974 CPN29H 10963480 Ki = 890 nM T62974 C6TVQ8 10964197 Ki = 316.23 nM T62974 CU70TI 10974426 Ki = 260 nM T62974 CK5XB4 10974575 Ki = 1200 nM T62974 CXDG12 10996788 Ki < 100 nM T62974 CJAH75 11050695 Ki = 570 nM T62974 C6AW0M 11112736 Ki = 9800 nM T62974 C5JX9W 11125276 Ki = 360 nM T62974 CK1RX4 11136828 Ki = 316.23 nM T62974 CR1JP9 11147505 Ki < 100 nM T62974 C1I9EX 11159133 IC50 = 3 nM T62974 C7REL4 11170698 IC50 = 1.8 nM T62974 CIEM12 11170867 IC50 = 453 nM T62974 CW2JA8 11182381 IC50 = 2.2 nM T62974 CE3GC2 11205475 IC50 = 0.7 nM T62974 CXI32T 11205496 IC50 = 0.88 nM T62974 C2RNJ5 11205515 IC50 = 1.1 nM T62974 CUT8Z0 11240205 IC50 = 1.8 nM T62974 CK78SD 11240206 IC50 = 1.3 nM T62974 C67WXD 11274767 IC50 = 0.51 nM T62974 COK06N 11320738 IC50 = 2.1 nM T62974 C5D6AM 11332138 IC50 = 0.98 nM T62974 C5PAN4 11343811 IC50 = 4.3 nM T62974 CLQ53A 11355270 IC50 = 3.5 nM T62974 CQ0UC7 11378229 IC50 = 41 nM T62974 CC09ZU 11378299 IC50 = 2 nM T62974 CG7PT9 11389178 IC50 = 1.5 nM T62974 CFJD72 11423410 IC50 = 1.1 nM T62974 C4S2HG 11434734 IC50 = 4 nM T62974 C3T6XG 11442741 Ki = 1.2 nM T62974 C6XHC3 11457491 IC50 = 1.2 nM T62974 CJ5A9B 11457521 IC50 = 1.1 nM T62974 CMA8C7 11468709 IC50 = 3.5 nM T62974 CG8A0J 11468887 IC50 = 1.3 nM T62974 CZ3N5J 11468916 IC50 = 1 nM T62974 CORY59 11480246 IC50 = 0.55 nM T62974 C63QMX 11535351 IC50 = 214 nM T62974 C0R6TS 11548587 IC50 = 440 nM T62974 CF6K7M 11563877 IC50 = 100 nM T62974 CS68YA 11642413 IC50 = 430 nM T62974 CZHN61 11678313 IC50 > 10000 nM T62974 CW65KY 11705763 Ki = 800 nM T62974 CN63YV 11787877 IC50 = 9.5 nM T62974 CR6UF9 11788180 IC50 = 3.5 nM T62974 CK7BN1 11800917 Ki = 96 nM T62974 CK4U8N 11804376 IC50 = 1000 nM T62974 C9XH7F 11815114 Ki < 100 nM T62974 CUI15C 11828523 IC50 = 53 nM T62974 CRA01O 11845058 IC50 = 494 nM T62974 C8X3CL 11845059 IC50 > 1000 nM T62974 CO3HT9 11847587 IC50 = 872 nM T62974 CAD8P9 11848624 Ki > 10000 nM T62974 CM49QW 11848625 Ki > 10000 nM T62974 CEBA46 11848626 Ki > 10000 nM T62974 CCT5G7 11848677 Ki > 10000 nM T62974 CMR10F 11848679 Ki > 10000 nM T62974 C9QDX3 11848833 Ki > 10000 nM T62974 CL6B5X 11848835 Ki > 10000 nM T62974 CW7I8U 13690207 IC50 = 3 nM T62974 C8OU7I 15429504 IC50 = 406 nM T62974 CEO3F0 15585102 IC50 = 8.2 nM T62974 CC2YJ8 16062553 Ki > 10000 nM T62974 C3H1RT 16062555 Ki > 10000 nM T62974 C1LH5T 16062816 Ki > 10000 nM T62974 C1GKF8 16130982 IC50 = 2.3 nM T62974 C2TRA5 16144717 IC50 = 605 nM T62974 CW20OC 16144977 IC50 = 1000 nM T62974 CS6A3Z 16145268 IC50 = 1000 nM T62974 CN3LS1 16145579 IC50 = 1000 nM T62974 C72MUC 16146425 IC50 = 312 nM T62974 CD91IL 16148220 IC50 = 2844 nM T62974 C59OUC 16148481 Ki < 79.43 nM T62974 CJG1X9 16148596 Ki < 1 nM T62974 CNY09C 16148922 Ki < 1000 nM T62974 CP0DC8 16149640 Ki < 0.631 nM T62974 CDPC19 16149975 Ki < 3.981 nM T62974 C0SE6V 16150676 Ki < 0.1995 nM T62974 CSP6A9 16150915 Ki < 0.1 nM T62974 C6N7SR 16151159 Ki < 1.995 nM T62974 C2B9IL 16151570 IC50 = 932 nM T62974 CQM8J1 16151781 IC50 = 1.2 nM T62974 CM8UF7 16151826 IC50 = 562 nM T62974 CJ7UT6 16151923 IC50 = 8.8 nM T62974 CIM03U 16152257 IC50 = 1.9 nM T62974 CU7X6V 16153077 IC50 = 0.9 nM T62974 CK4O1V 16153193 IC50 = 1.2 nM T62974 C16LMW 16153418 IC50 = 2.4 nM T62974 CO0LG7 16154000 IC50 = 2.1 nM T62974 CX4RM8 16154096 IC50 = 1.6 nM T62974 COYU86 16156815 Ki < 1000 nM T62974 CI3FW1 16157160 IC50 = 1000 nM T62974 C7GN0S 16157479 Ki < 0.1995 nM T62974 CQL5O0 16181427 IC50 > 1000 nM T62974 C2CUY9 16181428 IC50 > 1000 nM T62974 CUH8D7 16737812 IC50 = 129 nM T62974 C8QIT3 16737813 IC50 = 75 nM T62974 CNP36U 16737814 IC50 = 3.3 nM T62974 C7Q6JL 16738359 IC50 = 73 nM T62974 CJ9K1C 24740750 Ki > 10000 nM T62974 CS6VO9 24740751 Ki > 10000 nM T62974 CA4K0B 24740752 Ki > 10000 nM T62974 C4N3AX 24740753 Ki > 10000 nM T62974 COQU12 24740861 Ki > 10000 nM T62974 CAD4S1 24740862 Ki > 10000 nM T62974 C67YVI 24740863 Ki > 10000 nM T62974 CO0IF5 24740864 Ki > 10000 nM T62974 C6F1RZ 24777672 IC50 = 141 nM T62974 C5GZO7 24858018 IC50 = 0.9 nM T62974 CV1U7H 24858920 IC50 = 1 nM T62974 C0UB7K 24859055 IC50 = 2.6 nM T62974 CQCW58 24859056 IC50 = 1.3 nM T62974 CT6J2A 24859195 IC50 = 0.7 nM T62974 CUDV69 24859196 IC50 = 4.5 nM T62974 C45NYA 24859341 IC50 = 3.25 nM T62974 C4AB6I 24859342 IC50 = 3.1 nM T62974 CH50QU 24859494 IC50 = 1.9 nM T62974 C8L2KJ 24859495 IC50 = 6 nM T62974 CDS6W5 24859645 IC50 = 2 nM T62974 CHF20D 24859646 IC50 = 3 nM T62974 CKH2R4 24859787 IC50 = 1.5 nM T62974 CT1BM6 24859788 IC50 = 5 nM T62974 C2IKX3 24859919 IC50 = 4.4 nM T62974 C5OQ2X 24859920 IC50 = 2.7 nM T62974 CSZ73L 24860057 IC50 = 2.6 nM T62974 C36ZHQ 24860058 IC50 = 2.2 nM T62974 CVL48C 24860201 IC50 = 1.6 nM T62974 C20ZFS 24860202 IC50 = 1.4 nM T62974 C3C0KP 24894134 EC50 > 50000 nM T62974 CI8BZ6 24936235 Ki = 3200 nM T62974 CHKC79 25187396 IC50 = 7 nM T62974 C4YXJ1 25187398 IC50 = 8.1 nM T62974 CO9PI7 25187400 IC50 = 1.3 nM T62974 C8C9PL 25187679 IC50 = 2.3 nM T62974 C9ECD8 25187681 IC50 = 161 nM T62974 C43OES 25187683 IC50 = 14 nM T62974 CNTB73 25187685 IC50 = 6.9 nM T62974 C1IUQ2 25187953 IC50 = 2.1 nM T62974 CQ3F8L 25187955 IC50 = 35 nM T62974 CS2ZV1 25188218 IC50 = 14 nM T62974 CLI2U1 25188220 IC50 = 1 nM T62974 CNDU95 25188496 IC50 = 2.4 nM T62974 C7KF8N 25188776 IC50 = 56 nM T62974 CCHN50 25188780 IC50 = 7 nM T62974 C3T8DA 25189052 IC50 = 4.4 nM T62974 CI21ED 25189054 IC50 = 59 nM T62974 C97LHK 25189325 IC50 = 2.4 nM T62974 CEG4J0 25189327 IC50 = 17 nM T62974 CSQH26 42637069 IC50 = 95 nM T62974 CJ1S9K 42637136 IC50 = 525 nM T62974 C3NYM8 42637137 IC50 > 1000 nM T62974 CJ47CL 42637210 IC50 > 1000 nM T62974 CR3A8Q 42637283 IC50 > 1000 nM T62974 CENZ47 42637363 IC50 = 250 nM T62974 CX0JC7 42637503 IC50 = 27 nM T62974 C90LHS 42637563 IC50 = 266 nM T62974 C80WBK 42637632 IC50 = 270 nM T62974 CR49YE 42637984 IC50 > 1000 nM T62974 CEFO24 42638065 IC50 > 1000 nM T62974 CF5JK4 42638066 IC50 = 252 nM T62974 CHY04A 44290718 IC50 > 100 nM T62974 C16BKW 44290734 IC50 = 7 nM T62974 CW76YB 44290735 IC50 = 49.5 nM T62974 CA6IS7 44290766 IC50 > 100 nM T62974 C6BZ1J 44298104 Ki > 1000 nM T62974 CCXL10 44298113 Ki = 301 nM T62974 CB9JK1 44298131 Ki > 1000 nM T62974 CJ5WL8 44298155 Ki > 1000 nM T62974 CHL57J 44298156 Ki > 1000 nM T62974 CP61LB 44298165 Ki > 1000 nM T62974 CM0B6J 44298166 Ki > 1000 nM T62974 C8XZR7 44298169 Ki > 1000 nM T62974 C0DPX7 44298171 Ki = 1570 nM T62974 C62OEU 44298177 Ki > 1000 nM T62974 CS9JW8 44298178 Ki > 1000 nM T62974 C20MBI 44298179 Ki = 847 nM T62974 C3QBP0 44298188 Ki = 176 nM T62974 C1R3QD 44298189 Ki = 436 nM T62974 C5RJ7U 44298195 Ki > 1000 nM T62974 C8N3EJ 44298197 Ki > 1000 nM T62974 C1R2SL 44298204 IC50 = 800 nM T62974 CZU05A 44298214 Ki > 1000 nM T62974 CQUS98 44298218 Ki > 1000 nM T62974 COTK07 44298219 Ki > 1000 nM T62974 CAJO07 44298231 Ki = 728 nM T62974 C9S4IX 44298232 Ki = 672 nM T62974 CB1A3K 44298235 Ki = 1040 nM T62974 C2TQ1V 44298248 Ki > 1000 nM T62974 C3WFV5 44298250 Ki = 3310 nM T62974 CL2P9B 44298251 IC50 = 100 nM T62974 CMO1Q9 44298441 Ki > 1000 nM T62974 C8Y9ZP 44298443 Ki = 1590 nM T62974 CUSR45 44298468 Ki > 1000 nM T62974 C8EN2H 44298469 Ki > 1000 nM T62974 CWE7Q0 44298482 IC50 > 1000 nM T62974 CF69PL 44298522 Ki > 1000 nM T62974 CRQJ98 44308836 Ki = 2480 nM T62974 CRFM02 44308969 Ki = 2000 nM T62974 C40MJU 44308970 Ki = 1.76 nM T62974 C9KR7Q 44309052 Ki = 2176 nM T62974 C4YG1S 44311590 IC50 > 1000 nM T62974 CY0OV9 44311591 IC50 = 267 nM T62974 C29GQB 44311601 IC50 = 1.7 nM T62974 CC8DS0 44311602 IC50 > 1000 nM T62974 C5KST2 44311690 IC50 > 1000 nM T62974 C6N4MH 44311691 IC50 > 10000 nM T62974 CIR4G6 44311695 IC50 > 10000 nM T62974 CTG6X5 44311696 IC50 > 1000 nM T62974 C7Y8SF 44311697 IC50 > 1000 nM T62974 CK52MY 44311702 IC50 > 10000 nM T62974 CX39CV 44311703 IC50 > 1000 nM T62974 C5RM2A 44311730 IC50 > 1000 nM T62974 CBG70T 44311731 IC50 > 1000 nM T62974 CQH20F 44311765 IC50 > 10000 nM T62974 CZG4K6 44311836 IC50 = 487 nM T62974 CWNP79 44311837 IC50 > 1000 nM T62974 CEMH98 44311848 IC50 > 1000 nM T62974 CWSF38 44311868 IC50 > 1000 nM T62974 C2T0YP 44311869 IC50 > 10000 nM T62974 C1ONB3 44311870 IC50 > 1000 nM T62974 CXM6D3 44311888 IC50 > 1000 nM T62974 C1LQN0 44311889 IC50 > 1000 nM T62974 C1GY0F 44311912 IC50 > 1000 nM T62974 C14DIH 44311913 IC50 > 1000 nM T62974 C1X4TI 44311914 IC50 = 1.3 nM T62974 C74BDM 44311936 IC50 > 1000 nM T62974 C64WAE 44311958 IC50 > 1000 nM T62974 CFT90E 44311959 IC50 > 1000 nM T62974 C3PQD0 44311960 IC50 > 1000 nM T62974 C3WFS2 44311993 IC50 > 1000 nM T62974 CS7PB4 44312258 IC50 > 10000 nM T62974 C5PE1D 44325273 IC50 = 41 nM T62974 C1P0QV 44332931 Ki > 10000 nM T62974 CX1Y9V 44361984 Ki = 71000 nM T62974 C6UV4B 44362068 Ki = 50 nM T62974 CHP41F 44363816 Ki = 83 nM T62974 CH2DN4 44367916 IC50 > 1000 nM T62974 CM9YQ0 44367953 IC50 = 30 nM T62974 C5W4YL 44368019 IC50 = 14 nM T62974 CO6ZJ9 44368020 IC50 = 61 nM T62974 CQ5T1D 44368043 IC50 = 9.8 nM T62974 C1SWO5 44368044 IC50 = 21 nM T62974 C29EZK 44368080 IC50 = 1.8 nM T62974 C9ZW6U 44368093 IC50 = 11.8 nM T62974 C71URM 44368094 IC50 = 9.2 nM T62974 CC1ZP9 44368109 IC50 > 1000 nM T62974 CQ7OP1 44368112 IC50 = 8.7 nM T62974 C0EW4I 44368117 IC50 = 12 nM T62974 C6TNZ9 44368144 IC50 = 105 nM T62974 C53IAG 44368153 IC50 = 0.53 nM T62974 CKU8J7 44368156 IC50 = 0.7 nM T62974 CR12GB 44368157 IC50 = 1.8 nM T62974 C50DMO 44368226 IC50 = 6.9 nM T62974 CN31HS 44368398 IC50 = 24 nM T62974 C2RC0P 44368406 IC50 = 6.5 nM T62974 CB1HC8 44368422 IC50 = 429 nM T62974 C27DLY 44368489 IC50 = 80 nM T62974 CWHK38 44377332 Ki > 10000 nM T62974 CVH1O7 44377366 Ki > 5000 nM T62974 CRC2N1 44377555 Ki = 7200 nM T62974 CS1WT5 44377591 Ki > 10000 nM T62974 C3LUY8 44377623 Ki > 10000 nM T62974 CQD0P4 44377645 Ki > 5000 nM T62974 CWNF42 44385504 Ki = 3970 nM T62974 CAFD79 44385508 Ki > 10000 nM T62974 CHY14B 44385591 Ki > 10000 nM T62974 CJQI19 44385652 Ki = 7090 nM T62974 CG12HD 44385712 Ki = 5920 nM T62974 C8MU5C 44385757 Ki > 10000 nM T62974 C0LRT9 44386389 Ki = 6660 nM T62974 C1EVK8 44387399 Ki > 1000 nM T62974 C6U9VC 44388027 IC50 > 1000 nM T62974 C2IW5J 44388028 IC50 > 1000 nM T62974 C27ANT 44388029 IC50 = 611 nM T62974 CHQK20 44388035 IC50 > 1000 nM T62974 CI9XS1 44388036 IC50 > 1000 nM T62974 CD4BX6 44388037 IC50 = 215 nM T62974 CDS08Z 44388038 IC50 > 1000 nM T62974 CZA03Y 44388040 IC50 > 1000 nM T62974 C21WBR 44388043 IC50 > 1000 nM T62974 C7VK6B 44388052 IC50 > 1000 nM T62974 CT93BI 44388060 IC50 > 1000 nM T62974 C4E5VS 44388061 IC50 > 1000 nM T62974 C7P5RO 44388066 IC50 > 1000 nM T62974 C7T8IY 44388069 IC50 > 1000 nM T62974 C2TWO3 44388070 IC50 > 1000 nM T62974 CDBE87 44388075 IC50 > 1000 nM T62974 C25GWK 44388078 IC50 > 1000 nM T62974 CT93LV 44388079 IC50 > 1000 nM T62974 CX54SC 44388083 IC50 > 1000 nM T62974 C2C0RU 44388084 IC50 > 1000 nM T62974 C5SMA2 44388085 IC50 > 1000 nM T62974 C26OCG 44388086 IC50 > 1000 nM T62974 C8SR2O 44388087 IC50 > 1000 nM T62974 CHL5T1 44388088 IC50 > 1000 nM T62974 C4VNC2 44388089 IC50 > 1000 nM T62974 C1IH3T 44388090 IC50 > 1000 nM T62974 CNC91I 44388093 IC50 > 1000 nM T62974 CN45OF 44388095 IC50 = 700 nM T62974 C82HJL 44388104 IC50 > 1000 nM T62974 CV6T2H 44388105 IC50 > 1000 nM T62974 CLC0N2 44388106 IC50 > 1000 nM T62974 C0VO1K 44388107 IC50 > 1000 nM T62974 CM5O3B 44388108 IC50 > 1000 nM T62974 CAF02P 44388109 IC50 = 99 nM T62974 C23XBM 44388110 IC50 > 1000 nM T62974 CPX74G 44388112 IC50 > 1000 nM T62974 CG9SA3 44388114 IC50 = 772 nM T62974 C2C4MH 44388116 IC50 > 1000 nM T62974 CW1EL5 44388118 IC50 > 1000 nM T62974 CN0K3V 44388119 IC50 > 1000 nM T62974 CE8DH4 44388120 IC50 > 1000 nM T62974 C1A0OY 44388121 IC50 = 562 nM T62974 CS53NP 44388122 IC50 > 1000 nM T62974 CX67WG 44388123 IC50 = 435 nM T62974 CB50EK 44388124 IC50 = 660 nM T62974 C9SN1X 44388132 IC50 > 1000 nM T62974 C6W4YT 44388133 IC50 > 1000 nM T62974 CMTN20 44388134 IC50 > 1000 nM T62974 CAK42W 44388135 IC50 > 1000 nM T62974 CTW48B 44388136 IC50 > 1000 nM T62974 C4P1AS 44388137 IC50 > 1000 nM T62974 CEAZ82 44388138 IC50 > 1000 nM T62974 C1KMT8 44397389 Ki = 74 nM T62974 CN6Z8C 44397648 Ki = 130 nM T62974 CRW0M6 44397706 Ki = 140 nM T62974 CM1R8X 44400000 IC50 > 10000 nM T62974 CP89CS 44400135 IC50 = 300 nM T62974 C1BY2P 44444935 IC50 = 412 nM T62974 CH17TI 44560858 IC50 = 349 nM T62974 C2AZY7 44560859 IC50 = 287 nM T62974 C2I8NB 44560860 IC50 > 1000 nM T62974 C4XRT0 44560861 IC50 > 1000 nM T62974 C21TZI 44560862 IC50 > 1000 nM T62974 C2YM5N 44560863 IC50 > 1000 nM T62974 CS39FB 44560864 IC50 = 296 nM T62974 CU3FD2 44560865 IC50 = 715 nM T62974 C8IKU1 44560866 IC50 > 1000 nM T62974 CTQ83Z 44560867 IC50 = 116 nM T62974 CQC29N 44560868 IC50 = 908 nM T62974 C47MDA 44560869 IC50 = 479 nM T62974 CHAJ41 44560870 IC50 = 136 nM T62974 CT0A9U 44560871 IC50 = 831 nM T62974 CM0T9R 44560872 IC50 > 1000 nM T62974 CO2J6R 44560873 IC50 = 728 nM T62974 CKQD64 44560874 IC50 > 1000 nM T62974 CEK26Y 44560875 IC50 > 1000 nM T62974 CBL1P7 44560876 IC50 > 1000 nM T62974 CY47DM 44560877 IC50 = 800 nM T62974 C5OZD1 44560878 IC50 = 551 nM T62974 CFT47C 44560898 IC50 > 1000 nM T62974 CAO7R0 44560899 IC50 = 883 nM T62974 C80ZCF 44560900 IC50 = 813 nM T62974 CATH94 44560901 IC50 = 287 nM T62974 C2AXG6 44560902 IC50 = 905 nM T62974 COQ9W7 44560903 IC50 > 1000 nM T62974 CLZ23V 44560904 IC50 > 1000 nM T62974 C0OKG2 44560905 IC50 > 1000 nM T62974 CPIW17 44560906 IC50 > 1000 nM T62974 CFR3Y5 44560907 IC50 > 1000 nM T62974 CS85LR 44560908 IC50 = 455 nM T62974 C6K1FI 44577218 IC50 = 214 nM T62974 CAJ15T 44577219 IC50 = 115 nM T62974 CQD56E 44577220 IC50 = 296 nM T62974 CV18IC 44577221 IC50 = 174 nM T62974 C4NG5O 44820544 Ki = 690 nM T62974 CF5I4L 44820545 Ki = 160 nM T62974 CKRO61 44820563 Ki = 26 nM T62974 CTSR92 44820569 Ki = 19 nM T62974 CLJD09 45102042 IC50 > 10000 nM T62974 C63YJS 45139239 IC50 > 1000 nM T62974 C63XPN 45267999 IC50 > 1000 nM T62974 CF09UA 45268875 IC50 = 45 nM T62974 C2PNH4 45272264 IC50 > 1000 nM T62974 CFL9K7 45273129 IC50 = 296 nM T62974 C9Z4MR 45273130 IC50 > 1000 nM T62974 C4RGN0 45273131 IC50 = 71 nM T62974 CH18QA 46882131 Ki > 10000 nM T62974 CBZ3T9 46882132 Ki > 10000 nM T62974 C6KBJ2 46882133 Ki > 10000 nM T62974 CNL16U 46882180 Ki > 10000 nM T62974 CCX75M 46882181 Ki > 10000 nM T62974 C2BOJ6 46882182 Ki > 10000 nM T62974 C9ASC1 46882224 Ki > 10000 nM T62974 CB38SE 46882225 Ki > 10000 nM T62974 CP2N1U 46882226 Ki > 10000 nM T62974 CJ3Q6B 46882227 Ki > 10000 nM T62974 CRYQ47 46882445 Ki > 10000 nM T62974 CRZ1B0 46882446 Ki > 10000 nM T62974 CNEZ46 46882447 Ki > 10000 nM T62974 C8D1OR 46882448 Ki > 10000 nM T62974 CZ0G2R 46882449 Ki > 10000 nM T62974 CR37UF 46882513 Ki > 10000 nM T62974 CF3L8U 46882514 Ki > 10000 nM T62974 C91WKZ 46882515 Ki > 10000 nM T62974 CX21JH 46882516 Ki > 10000 nM T62974 CBJ92C 46882517 Ki > 10000 nM T62974 C8N3KX 46882577 Ki > 10000 nM T62974 CAH31I 46882578 Ki > 10000 nM T62974 CD2NL0 46882579 Ki > 10000 nM T62974 C9B0DF 46882620 Ki > 10000 nM T62974 CJ8I4L 46882621 Ki > 10000 nM T62974 C2YMA7 46882622 Ki > 10000 nM T62974 CD0VH7 46882664 Ki > 10000 nM T62974 C50YRJ 46882665 Ki > 10000 nM T62974 CXFV62 46882666 Ki > 10000 nM T62974 CR07WV 46882667 Ki > 10000 nM T62974 CF1HC7 46882668 Ki > 10000 nM T62974 CVIU56 46882708 Ki > 10000 nM T62974 C8S4LN 46882709 Ki > 10000 nM T62974 CJ7GM9 46882746 Ki > 10000 nM T62974 C6OM5H 46882789 Ki > 10000 nM T62974 C5MV8K 46882790 Ki > 10000 nM T62974 C6RD3V 46882791 Ki > 10000 nM T62974 C1WUF9 46882831 Ki > 10000 nM T62974 C5LM3W 46882832 Ki > 10000 nM T62974 CU1D6I 46902023 IC50 = 4000 nM T62974 CG78MV 46919128 IC50 = 180 nM T62974 C84ZTC 49865341 IC50 = 412 nM T62974 C3VZ4U 49865342 IC50 > 1000 nM T62974 CGYR09 49865343 IC50 = 346 nM T62974 C35WID 49865344 IC50 = 249 nM T62974 C0RK7G 49865345 IC50 = 1000 nM T62974 C4YLM7 49865346 IC50 > 1000 nM T62974 CZ4RI1 49865347 IC50 > 1000 nM T62974 CQJP15 51003591 Ki = 4400 nM T62974 C9SNL1 52941607 IC50 > 10000 nM T62974 CO04IG 52943613 IC50 = 660 nM T62974 CVO9X2 52947330 IC50 = 720 nM T62974 C40ZRY 52948630 IC50 > 10000 nM T62974 CED3O6 53473658 IC50 = 25 nM T62974 CE7J0U 53473659 IC50 = 16 nM T62974 CY0G2K 53473744 IC50 = 12 nM T62974 CBQG96 53473824 IC50 = 12 nM T62974 CW53YV 53473917 IC50 > 1000 nM T62974 C87SME 53474004 IC50 > 1000 nM T62974 C7EO1Z 53474005 IC50 > 1000 nM T62974 CY3M2A 53474090 IC50 = 590 nM T62974 CM58UZ 56651206 IC50 = 1200 nM T62974 COBQ28 56651207 Ki = 580 nM T62974 CGKP76 56661222 Ki = 60 nM T62974 C3RWH0 56661224 Ki = 124 nM T62974 C9JHI4 56664813 Ki = 2 nM T62974 C3M6AT 56678313 Ki < 1 nM T62974 C05RSG 56681656 Ki = 700 nM T62974 C59PKT 56681657 Ki = 3.7 nM T62974 C4MT8I 56681776 IC50 = 100 nM T62974 C8ZW3O 56927659 IC50 = 384 nM T62974 CHK8T1 56945132 EC50 = 6.8 nM T62974 C73XBL 57384077 IC50 > 1000 nM T62974 C3KC9Z 57398462 IC50 = 2.5 nM T62974 CTVI05 70683416 IC50 = 214 nM T62974 CV42WQ 70689221 IC50 = 6.9 nM T62974 C3P0AN 70689413 IC50 > 1000 nM T62974 CP58HL 70689414 IC50 > 1000 nM T62974 CB14OW 70689415 IC50 > 1000 nM T62974 CNZC97 70689723 IC50 = 63 nM T62974 C2WQM9 70691295 IC50 > 1000 nM T62974 C5E8MY 70693613 IC50 = 373 nM T62974 C3TZ9U 70695246 IC50 = 932 nM T62974 C34XGS 70695722 IC50 > 1000 nM T62974 CIPF50 70695723 IC50 > 1000 nM T62974 CF08XL 71458043 Ki = 7200 nM T62974 CU82HG 71460000 IC50 > 1000 nM T62974 CPC69G 71461645 Ki > 10000 nM T62974 CLAV92 71461684 IC50 > 1000 nM T62974 C1NZU3 71461685 IC50 > 10000 nM T62974 CI0GU8 71660496 IC50 > 48500 nM T62974 CFKH42 71717904 IC50 = 1000 nM T62974 CGDO59 72947672 Ki = 1.77 nM T62974 CW83DK 73213196 Ki > 10000 nM T62974 CIO28F 73345407 Ki = 1000 nM T62974 CMN6X8 73345525 IC50 = 5.4 nM T62974 C70XZC 73345528 IC50 = 1.2 nM T62974 CXGJ67 73345700 IC50 = 729 nM T62974 CV23JS 73345701 IC50 = 1033 nM T62974 C81UME 73345740 Ki > 1000 nM T62974 CX5VM1 73346900 IC50 > 10000 nM T62974 CA3MU5 73346903 IC50 = 3.5 nM T62974 C62NFY 73346927 Ki = 575 nM T62974 CK64MX 73346930 Ki = 1000 nM T62974 C15CAN 73346972 Ki > 1000 nM T62974 CD09FU 73347225 Ki = 2880 nM T62974 CI4L6W 73347226 Ki = 682 nM T62974 CGM61R 73348311 Ki > 10000 nM T62974 CN1FD2 73348312 Ki > 10000 nM T62974 C01GIQ 73348427 Ki = 1000 nM T62974 C7Y9ZT 73348428 Ki = 1000 nM T62974 CFLT50 73348719 IC50 = 61.8 nM T62974 C75NBQ 73348741 Ki = 145 nM T62974 C5MNX3 73348742 Ki > 1000 nM T62974 CL94MY 73350006 Ki = 1000 nM T62974 C0N6XK 73350010 Ki = 1000 nM T62974 CTV30F 73350011 Ki = 1000 nM T62974 CF2AK4 73350012 Ki = 1000 nM T62974 CK9CS4 73351516 Ki = 1000 nM T62974 CNY13O 73351517 Ki = 1000 nM T62974 CUN6L1 73351622 IC50 = 41 nM T62974 CC98JE 73351624 IC50 = 1.4 nM T62974 CWUH52 73351718 Ki = 1246 nM T62974 CS9I4W 73351829 Ki > 1000 nM T62974 CF70XH 73351873 IC50 > 1000 nM T62974 C0KJ6N 73352984 Ki = 80 nM T62974 CFB54J 73352985 Ki = 1000 nM T62974 CKFV85 73353009 Ki = 987 nM T62974 CC45AV 73353272 IC50 = 337 nM T62974 C41OCY 73353278 IC50 = 35.9 nM T62974 CW54CU 73353340 IC50 > 1000 nM T62974 CL7DT2 73354494 Ki = 1000 nM T62974 CA48EL 73354535 Ki > 1000 nM T62974 CFK7Z3 73354633 IC50 = 3.5 nM T62974 C1UYL2 73354783 IC50 = 346 nM T62974 CG1CX0 73354798 IC50 > 100 nM T62974 CIVZ67 73354818 Ki = 895 nM T62974 CGCE64 73354819 Ki = 888 nM T62974 C1Y0CI 73356066 Ki = 1000 nM T62974 C52JAS 73356068 Ki = 1000 nM T62974 CN5LG8 73356069 Ki = 1000 nM T62974 C9GKV2 73356181 IC50 = 2.3 nM T62974 C7XFB6 73356331 IC50 = 4.11 nM T62974 CI02SE 73356366 Ki = 1640 nM T62974 CW8L6C 76310862 IC50 > 1000 nM T62974 CHV6K7 76314485 IC50 = 5.4 nM T62974 C0PR3Y 76314486 IC50 > 1000 nM T62974 C94BWD 76314487 IC50 = 2.8 nM T62974 C25XKO 76314488 IC50 = 0.9 nM T62974 CS54IV 76321777 IC50 = 4 nM T62974 C94OAT 76321778 IC50 = 1.2 nM T62974 CU1IR8 76325402 IC50 = 3.7 nM T62974 CL09JQ 86279005 IC50 > 10000 nM T62974 C3JOS4 86292350 EC50 = 1.2 nM T62974 CVLE34 86293506 EC50 = 0.4 nM T62974 C15VTO 86294248 EC50 = 0.4 nM T62974 C2BAV8 90644981 Ki = 1089 nM T62974 CI58FM 90663867 IC50 = 837 nM T62974 CK62FO 90663868 IC50 > 1000 nM T62974 C7AFD4 90663869 IC50 = 482 nM T62974 C94XTF 90663872 IC50 > 1000 nM T62974 CA7W0U 90663873 IC50 = 797 nM T62974 C4EG8T 90663874 IC50 = 823 nM T62974 CW21UO 90663875 IC50 = 356 nM T62974 C7Q4PD 90665458 Ki = 20000 nM T62974 CR43ZL 90665459 Ki = 4900 nM T62974 CLK7C3 90665460 Ki = 7200 nM T62974 CZ0UC6 90665461 Ki = 10000 nM T62974 C0IBJ6 90665462 Ki = 21000 nM T62974 CPX0C9 90665463 Ki = 12000 nM T62974 C3UVC8 91936728 IC50 > 1000 nM T62974 CT3UP7 91936729 IC50 = 523 nM T62974 CD2E4L 101941290 IC50 = 1000 nM T62974 C9KB3W 117711399 EC50 = 4.3 nM T62974 CTH52C 118718416 Ki < 0.3162 nM T62974 CKQ4P6 118718462 IC50 = 1172 nM T62974 C1Z7UJ 118718463 Ki < 1000 nM T62974 CPYA80 118718465 IC50 = 1000 nM T62974 CR61UD 118718466 IC50 = 1000 nM T62974 CW64XN 118718500 IC50 = 1000 nM T62974 CB4D5T 118718501 IC50 = 632 nM T62974 CW5HG2 118718502 IC50 = 1000 nM T62974 CC36KP 118718503 IC50 = 1000 nM T62974 C7FIQ1 118718504 IC50 = 1000 nM T62974 CNBY57 118718505 IC50 = 3007 nM T62974 CPY4Q5 118718506 IC50 = 757 nM T62974 CO13JR 118718507 IC50 = 1000 nM T62974 CLFJ60 118718508 IC50 = 1000 nM T62974 C13YUH 118718509 IC50 = 1000 nM T62974 CP2O7U 118718510 IC50 = 1000 nM T62974 CLDZ63 118718511 IC50 = 1000 nM T62974 CYQ7X2 118718854 IC50 = 31 nM T62974 CA6C4T 118719101 IC50 = 2.3 nM T62974 CDZ3H4 118719196 IC50 = 2.4 nM T62974 CQRO32 118719197 IC50 = 5.6 nM T62974 CGXH91 118719198 IC50 = 3.2 nM T62974 C1QJX7 118719199 IC50 = 2.6 nM T62974 C0GLC8 118719200 IC50 = 153 nM T62974 C40NGQ 118719201 IC50 = 133 nM T62974 CK2W9T 118719202 IC50 = 5.2 nM T62974 CW4AT0 118719275 IC50 = 5.4 nM T62974 C5VWI1 118719303 IC50 = 1000 nM T62974 CS12JW 122179457 IC50 = 3200 nM T62974 CNGQ19 122179477 IC50 > 100000 nM T62974 C9B4DJ 122181226 Ki = 5400 nM T62974 CH1P7L 122181227 Ki = 1900 nM T62974 C6M3TH 127032865 Ki = 7090 nM T62974 CB5Q9D 127032866 Ki = 1170 nM T62974 CUO25F 127032867 Ki = 2020 nM T62974 CF1T6D 127033186 Ki = 2050 nM T62974 CE79SV 138377584 IC50 > 10000 nM T62974 C9CEY3 145949026 Ki = 1.34 nM T62974 CP0WF8 155510657 IC50 > 100000 nM T62974 C0I2UD 155513010 Ki > 10000 nM T62974 CV2BZ9 155516168 Ki > 10000 nM T62974 C2OG9Y 155517592 Ki > 10000 nM T62974 C59SVW 155518749 Ki > 10000 nM T62974 C1BS2T 155519582 Ki = 1426 nM T62974 CHJO90 155524485 Ki > 10000 nM T62974 CW0XC1 155526536 IC50 = 103 nM T62974 CD73TA 155526663 IC50 > 100000 nM T62974 CGXE80 155528330 Ki = 6800 nM T62974 C9QIB6 155529288 Ki = 7200 nM T62974 CI9HE4 155532172 Ki < 10000 nM T62974 CYT0Z4 155532886 Ki > 10000 nM T62974 CKZ82R 155538553 Ki > 10000 nM T62974 C9XB6L 155539840 Ki > 100000 nM T62974 CVOW56 155541238 Ki > 10000 nM T62974 CBD2Q8 155541853 Ki = 2.41 nM T62974 C5RI8K 155541897 Ki = 21000 nM T62974 CIA72K 155543246 IC50 > 100000 nM T62974 CVR3U2 155546680 Ki = 1900 nM T62974 CY68DL 155546826 Ki = 4471 nM T62974 CGZY28 155549889 Ki > 100000 nM T62974 CLJU08 155550820 Ki = 20000 nM T62974 CI6E8B 155552577 Ki > 10000 nM T62974 C89BNQ 155553012 Ki = 2100 nM T62974 CX02AJ 155555535 Ki = 4803 nM T62974 CR1AY2 155557409 Ki = 2380 nM T62974 CD58IO 155558366 Ki = 2032 nM T62974 C6T0IB 155560534 Ki > 10000 nM T62974 C5RL2K 155565048 Ki = 5400 nM T62974 CN7CQ1 155567326 Ki > 10000 nM T62974 CE76TG 42637005 IC50 = 468 nM T62974 C6ELN4 42637006 IC50 = 329 nM T62974 CS73LG 42637433 IC50 > 1000 nM T62974 C6C3YF 45270549 IC50 > 1000 nM T62974 C9Y3BS 45270550 IC50 > 1000 nM T62974 CQC51Z 45270552 IC50 > 1000 nM T62974 CXE30U 45271377 IC50 > 1000 nM T62974 D01BWV 9802572 Ki = 7100 nM T62974 D01NID 44388055 IC50 > 1000 nM T62974 D02CQW 11847438 IC50 > 1000 nM T62974 D02NJV 44388048 IC50 = 932 nM T62974 D02OJQ 44388115 IC50 = 0.5 nM T62974 D02WOX 44388129 IC50 > 1000 nM T62974 D03DRL 44388045 IC50 = 417 nM T62974 D03SXC 44388041 IC50 > 1000 nM T62974 D03VHX 44388111 IC50 > 1000 nM T62974 D04EWA 44388034 IC50 > 1000 nM T62974 D04FPW 44388024 IC50 > 1000 nM T62974 D04ORV 44388047 IC50 = 0.6 nM T62974 D04QBM 5311374 Ki = 0.7 nM T62974 D05COQ 11847588 IC50 > 1000 nM T62974 D05XZA 44388071 IC50 > 1000 nM T62974 D06JWT 44388073 IC50 > 1000 nM T62974 D07DUF 44388130 IC50 > 1000 nM T62974 D07OSF 44388044 IC50 > 1000 nM T62974 D07WRP 15965425 Ki = 81 nM T62974 D09DAC 44388046 IC50 = 1.2 nM T62974 D09LHN 44311674 IC50 = 384 nM T62974 D0A0DO 44388056 IC50 > 1000 nM T62974 D0A1XX 44388113 IC50 = 418 nM T62974 D0BE3D 44388092 IC50 > 1000 nM T62974 D0C5RH 44388125 IC50 = 1.4 nM T62974 D0CC1P 44388042 IC50 > 1000 nM T62974 D0H0DC 44388051 IC50 = 786 nM T62974 D0H4WH 44388128 IC50 = 1.7 nM T62974 D0I9ME 44388074 IC50 > 1000 nM T62974 D0J5OY 44388022 IC50 = 3.3 nM T62974 D0M5LA 44388050 IC50 > 1000 nM T62974 D0N2MA 44388103 IC50 > 1000 nM T62974 D0N4LH 44388065 IC50 > 1000 nM T62974 D0O4GU 44403230 Ki > 1000 nM T62974 D0P6ZZ 10581102 IC50 > 1000 nM T62974 D0R0OX 44388102 IC50 = 245 nM T62974 D0R4IS 44388131 IC50 > 1000 nM T62974 D0S7YR 44388059 IC50 > 1000 nM T62974 D0T5RO 16129706 Ki = 0.59 nM T62974 D0W0AF 44388072 IC50 = 226 nM T62974 D0WG0O 44388049 IC50 = 229 nM T62974 D0Z0OF 44388094 IC50 > 1000 nM T62974 D0Z1XY 44388064 IC50 > 1000 nM T62974 D0Z3LZ 44388023 IC50 = 1 nM T90818 D0V2GT 5311023 Ki = 84 nM T90818 C65NED 9573348 EC50 = 1000 nM T90818 CL57KJ 9707420 EC50 = 501.19 nM T90818 C2H5NY 9854861 Ki = 1.2 nM T90818 C3H7AS 9955930 Ki = 92 nM T90818 CH1Q6E 10008757 Ki > 3000 nM T90818 C6S2CB 25138123 IC50 = 2400 nM T90818 CMTA17 44542176 EC50 = 1258.93 nM T90818 COW17D 44542178 EC50 = 501.19 nM T90818 C7Q9PI 44542320 EC50 = 794.33 nM T90818 CY14UJ 44542322 EC50 = 398.11 nM T90818 C3ILH8 44542324 EC50 = 100 nM T90818 C8D4AT 44542326 EC50 = 199.53 nM T90818 CIRQ85 44542328 EC50 = 100 nM T90818 CB58DA 44542330 EC50 = 158.49 nM T90818 CS12HR 44542332 EC50 = 125.89 nM T90818 CY4L2G 53318788 IC50 = 0.79 nM T90818 CO72VY 60168134 EC50 = 1256 nM T90818 CW7KQ1 60168135 EC50 = 298 nM T90818 CH58GJ 71450762 Ki = 227 nM T90818 C6AV0I 71451611 EC50 = 1.7 nM T90818 C7K8BZ 71452593 Ki = 425 nM T90818 COM10Q 71454352 Ki = 142 nM T90818 CM31QR 71454353 Ki = 424 nM T90818 CL9E0V 71454357 Ki = 672 nM T90818 C8MP1A 71454358 Ki = 94 nM T90818 CHFO89 71454359 Ki = 417 nM T90818 C7ROU1 71456101 Ki = 117 nM T90818 CO07CE 71456102 Ki = 1620 nM T90818 C24UFT 71456103 Ki = 47 nM T90818 CL82IR 71456104 Ki = 9 nM T90818 C3SOE7 71457908 Ki = 136 nM T90818 CZ7C4L 71457909 Ki = 4 nM T90818 CJWQ68 71457910 Ki = 155 nM T90818 C3W7BS 71461185 Ki = 2015 nM T90818 C0VA5C 71463271 Ki = 141 nM T90818 C49KZP 71463273 Ki = 208 nM T90818 C1EGB8 71463275 Ki = 3196 nM T90818 CW9XZ8 71463276 Ki = 206 nM T90818 CA7S8C 71463277 Ki = 590 nM T90818 C75FXY 71463278 Ki = 4 nM T90818 CA7G4S 71463279 Ki = 22 nM T90818 CU9O4B 101493753 Ki = 0.53 nM T90818 CW3LH2 101882818 Ki = 1052 nM T90818 CW5H9D 101882819 Ki = 1426 nM T90818 CGQV37 101882820 Ki = 30 nM T90818 CA51CQ 118724536 Ki = 75 nM T90818 CR4MG1 118724537 Ki = 0.47 nM T90818 CBA2Z0 118724538 Ki > 5000 nM T90818 CL3T4A 118724539 Ki = 1694 nM T90818 CTHD48 118724540 Ki = 304 nM T90818 CZL32K 118724541 Ki > 5000 nM T90818 C5HNX2 118724542 Ki = 6616 nM T90818 C4AT2F 118724543 Ki = 2773 nM T90818 CE1NT2 118724544 Ki = 7579 nM T90818 CM3RN4 118724970 Ki = 2907 nM T90818 C5XD1N 118724971 Ki = 3220 nM T90818 C6M1AZ 118724972 Ki = 2682 nM T90818 CSF21L 118724973 Ki = 2223 nM T90818 CH4LB0 118724977 Ki = 405 nM T90818 C6GK5N 118724978 Ki = 1893 nM T90818 C9SN0M 118724979 Ki = 309 nM T90818 CH9GT5 118724980 Ki = 987 nM T90818 CHK0S7 118724981 Ki = 884 nM T90818 C1BVC2 118724982 Ki = 409 nM T90818 C76XZK 118724983 Ki = 3505 nM T90818 CG7SQ8 118724984 Ki = 84 nM T90818 CB3D6X 118724985 Ki = 465 nM T90818 CG04KW 118724986 Ki = 2757 nM T90818 CO69YD 118724987 Ki = 298 nM T90818 C72AKO 118724988 Ki = 330 nM T90818 C4CRS0 118724989 Ki = 129 nM T90818 CJIB02 118724990 Ki = 504 nM T90818 CD41AL 118724991 Ki = 454 nM T90818 C2DCZ3 118724992 Ki = 1513 nM T90818 C49HSM 118724993 Ki = 82 nM T90818 CE9ZS5 118724994 Ki = 205 nM T90818 CP2WY4 118724995 Ki = 910 nM T90818 C1TD6L 127030365 Ki = 41 nM T90818 C7YA8H 127030940 Ki = 27 nM T90818 C5PA2G 127041908 Ki = 1200 nM T90818 C62JIE 127042244 Ki > 3000 nM T90818 CNX9D2 136948074 Ki = 1620 nM T90818 CY35MT 136998789 Ki = 993 nM T90818 CBAP98 136998790 Ki = 2398 nM T90818 C8F9WQ 155515973 EC50 = 250 nM T90818 CF42WX 155520785 EC50 = 158.49 nM T90818 D01VSI 25240297 IC50 = 76 nM T90818 D08UWO 53320361 Ki = 43 nM T90818 D0JE3Z 16735569 IC50 = 1800 nM T17339 D0I2AN 86298439 IC50 = 2900 nM T17339 CKH70I 72705451 Ki = 150000 nM T17339 C0IJ2X 118737463 IC50 = 5700 nM T17339 CG0Z1I 137649766 Ki = 6900 nM T93283 C7GTI4 81312 IC50 > 500000 nM T93283 CFB8H3 96536 IC50 = 30000 nM T93283 CE0U1R 195023 IC50 = 142000 nM T93283 CEP2N4 242551 IC50 > 500000 nM T93283 CJR57B 4469578 IC50 = 4 nM T93283 CW9DQ2 4476325 IC50 = 6000 nM T93283 C0KAB3 9867336 IC50 = 1400 nM T93283 CIYE74 9881235 IC50 = 88000 nM T93283 CUJI84 9973036 IC50 = 9000 nM T93283 C3PB6D 10039105 IC50 = 14000 nM T93283 C2L3NF 10383023 IC50 = 21000 nM T93283 CIWE62 15341136 IC50 = 9300 nM T93283 CB9R2F 22988798 IC50 = 38000 nM T93283 C9LR1V 44296499 IC50 = 21000 nM T93283 C20DWM 44296500 IC50 = 11400 nM T93283 CFL2N8 44296527 IC50 = 6300 nM T93283 CIU45S 44296534 IC50 = 11000 nM T93283 C7N2KA 44296536 IC50 = 89000 nM T93283 C4R6WG 44309346 IC50 = 14000 nM T93283 C76YXK 44309396 IC50 = 8.6 nM T93283 C5XCT6 44336394 IC50 = 152000 nM T93283 CBM6E8 44336450 IC50 = 70000 nM T93283 C3P1KZ 44336452 IC50 = 67000 nM T93283 CBS80R 44336458 IC50 = 31000 nM T93283 C7RQ4C 44336463 IC50 = 37000 nM T93283 C58SWT 44336464 IC50 = 143000 nM T93283 CG0AV1 44336465 IC50 = 41000 nM T93283 CR32EI 44336472 IC50 = 100000 nM T93283 CAK08U 44336531 IC50 = 15000 nM T93283 CL2V8T 44336543 IC50 = 17000 nM T93283 C32ZLU 44336551 IC50 = 16000 nM T93283 CT31VP 44336553 IC50 = 36000 nM T93283 C98QZE 44336560 IC50 = 94000 nM T93283 C0VI7H 44336562 IC50 = 67000 nM T93283 CP1Z0W 49797574 IC50 = 1210 nM T93283 CK0X5J 49797575 IC50 = 25.7 nM T93283 CAJ35Z 49797576 IC50 = 1070 nM T93283 CZ7PV6 49797577 IC50 = 18 nM T93283 CI27BD 49797578 IC50 = 5 nM T93283 C3ETV8 49797579 IC50 = 198 nM T93283 D0N4XG 417214 IC50 = 34000 nM T75570 D0E6XR 3062316 IC50 = 0.5 nM T75570 D0OB0F 5328940 IC50 = 0.4 nM T75570 D03LWG 53235510 IC50 = 1100 nM T75570 D05PZB 135398495 IC50 = 1 nM T75570 D07EHV 44814409 IC50 > 10000 nM T75570 D0E0NM 25066467 IC50 = 1.5 nM T75570 D0E3TC 44259 IC50 = 2.35 nM T75570 D0G2QH 10297043 IC50 = 13.1 nM T75570 D0GP9Q 11973736 IC50 >= 2500 nM T75570 D0M0XB 10302451 IC50 = 0.7 nM T75570 D03BNU 59604787 IC50 > 10000 nM T75570 D0T3ME 156422 IC50 = 8900 nM T75570 CB1VW3 1400 IC50 = 36 nM T75570 CY13FW 644243 IC50 = 510 nM T75570 CR0DJ8 4078145 IC50 = 7700 nM T75570 CI80BK 9803350 IC50 = 20 nM T75570 CM2VB6 10100735 IC50 = 156000 nM T75570 C6DC8Q 10275163 IC50 = 10 nM T75570 C8RD3V 10301884 IC50 = 3 nM T75570 C5CBF9 10320381 IC50 = 10 nM T75570 CLAX64 10413508 IC50 = 30 nM T75570 CDQO71 10461517 IC50 = 110000 nM T75570 CJ5M1D 10482445 IC50 = 10 nM T75570 CACS26 11561968 Ki > 2000 nM T75570 CJV20L 11569758 IC50 = 4.1 nM T75570 CAJQ78 11584678 IC50 = 1.3 nM T75570 CU0E8O 11690457 Ki > 2000 nM T75570 CHL5W3 11712625 IC50 = 0.3 nM T75570 CZY05V 11719421 IC50 = 1.2 nM T75570 C73MLJ 16108977 IC50 = 8.7 nM T75570 C6TQ2O 16664354 Ki = 5.97 nM T75570 CY1E2N 16723801 IC50 = 30000 nM T75570 CG12OL 23518511 IC50 = 20 nM T75570 C6O8QY 23661616 IC50 = 4.8 nM T75570 CA3I4T 24753787 IC50 > 50000 nM T75570 CP1WR0 24795070 IC50 = 240 nM T75570 C2MUA7 24823072 IC50 = 110 nM T75570 CX94DT 24823073 IC50 = 22 nM T75570 CCFQ29 44187005 IC50 = 246 nM T75570 CH3J2E 44299176 IC50 = 40 nM T75570 C27GVO 44299203 IC50 = 160 nM T75570 CY6WC0 44299236 IC50 = 10 nM T75570 C3RG0C 44299304 IC50 = 20 nM T75570 CJM26I 44299321 IC50 = 10 nM T75570 C9UGL3 44299325 IC50 = 10 nM T75570 CJEZ96 44299338 IC50 = 40 nM T75570 C8XGN5 44299339 IC50 = 30 nM T75570 CNH34G 44299354 IC50 = 10 nM T75570 C82MSD 44299360 IC50 = 30 nM T75570 CJ3PF9 44313929 IC50 > 500000 nM T75570 CUV7K3 44313930 IC50 > 500000 nM T75570 CHK9N3 44313931 IC50 = 94500 nM T75570 CEKR19 44313990 IC50 > 500000 nM T75570 CD5PI9 44313997 IC50 = 2600 nM T75570 C0GH7J 44314372 IC50 > 500000 nM T75570 C5E4GK 44314373 IC50 > 500000 nM T75570 C3YD1G 44314380 IC50 = 303000 nM T75570 CPC68H 44314402 IC50 > 500000 nM T75570 C1L6MG 44444041 IC50 = 5.2 nM T75570 C3VRO9 44557921 IC50 > 10000 nM T75570 CYT37A 46232443 IC50 > 50000 nM T75570 C48ZVW 46232555 IC50 = 26000 nM T75570 CS9B1U 46232556 IC50 > 50000 nM T75570 CL0O4U 46911726 Ki = 24 nM T75570 CCN08S 46934144 IC50 = 38100 nM T75570 CG5IK8 52936268 IC50 > 100000 nM T75570 CEQN27 52936621 Ki > 1000 nM T75570 C2CT5J 53236670 IC50 = 7950 nM T75570 C3M6LV 53236671 IC50 > 100000 nM T75570 CZ5L6F 53239373 IC50 > 100000 nM T75570 C2WFI8 53239374 IC50 = 41800 nM T75570 C0ZHF8 53239375 IC50 = 85540 nM T75570 CD1EQ3 53239587 IC50 = 26940 nM T75570 C8NA4L 53384644 IC50 > 30000 nM T75570 CPHX64 57325478 IC50 > 50000 nM T75570 CQ9BW4 57325479 IC50 > 50000 nM T75570 C1JLW8 57332840 IC50 = 5560 nM T75570 CD01JZ 57332841 IC50 = 5110 nM T75570 CCFK37 57332844 IC50 = 5340 nM T75570 CK1SR7 57332969 IC50 = 2410 nM T75570 C5TRE2 57332970 IC50 = 2010 nM T75570 C46TJK 57332974 IC50 = 8820 nM T75570 C09ZJY 57333095 IC50 = 11100 nM T75570 CVK0G4 58056356 IC50 > 50000 nM T75570 C1MR8Q 60097495 IC50 > 1000 nM T75570 CE49GC 67098566 Ki = 79 nM T75570 CV63UL 67240318 IC50 > 10000 nM T75570 CAIO65 68796885 IC50 = 44 nM T75570 COU73Y 71226944 IC50 = 37 nM T75570 C40JOZ 71235465 IC50 = 73 nM T75570 C5ZKU7 71546969 IC50 = 284 nM T75570 C7ARI9 71547113 IC50 = 496 nM T75570 CDJY72 71568837 IC50 = 1800 nM T75570 C8CAG7 71578921 IC50 > 10000 nM T75570 C7E6YV 71720026 IC50 = 160.4 nM T75570 CGDB30 74538658 IC50 = 30 nM T75570 CPG3A5 86302574 IC50 > 30000 nM T75570 CQCX41 118737057 IC50 = 0.8 nM T75570 CKBP72 121231408 IC50 < 0.5 nM T75570 C81IFQ 122163152 IC50 > 100000 nM T75570 CCXA46 122190499 Ki = 470 nM T75570 C3PQ4W 122190505 Ki = 610 nM T75570 CN1DK0 122190507 Ki = 800 nM T75570 CD67LU 122705248 IC50 = 12 nM T75570 CX63VW 122705258 IC50 = 696 nM T75570 C76IKM 122705261 IC50 = 566 nM T75570 C8ALO2 124088839 IC50 = 344 nM T75570 C0HN2Y 127030123 IC50 = 22060 nM T75570 C7S9GI 127030124 IC50 > 31600 nM T75570 CHGN68 127030424 IC50 = 6210 nM T75570 CRV62L 127030425 IC50 > 31600 nM T75570 CF7JT8 127030426 IC50 > 31600 nM T75570 C5YCU2 127030427 IC50 > 31600 nM T75570 C0GES2 127031075 IC50 > 100000 nM T75570 CFJ32Y 127031076 IC50 > 100000 nM T75570 CC8V4J 127031368 IC50 = 27210 nM T75570 C78GYH 127031383 IC50 = 20430 nM T75570 C5WA9Z 127031384 IC50 = 31510 nM T75570 CD7LN1 127031385 IC50 = 8100 nM T75570 CI0VX4 127031386 IC50 = 12630 nM T75570 CO89TC 127031387 IC50 = 1020 nM T75570 CAM4S5 127031675 IC50 = 7070 nM T75570 C4QD0M 127031676 IC50 = 23110 nM T75570 C0LTC3 127031677 IC50 > 100000 nM T75570 CO1G2K 127032542 IC50 > 100000 nM T75570 C12IOL 127033165 IC50 > 31600 nM T75570 C5RO0L 127033758 IC50 > 100000 nM T75570 CD04YX 127034308 IC50 > 31600 nM T75570 CG8DA9 127045861 IC50 > 100000 nM T75570 CC4ND8 127046862 IC50 > 100000 nM T75570 CO25WH 127052538 IC50 = 71 nM T75570 C8F0DQ 129909860 IC50 = 4 nM T75570 CLCO61 135398510 IC50 = 1.4 nM T75570 CAW0E4 136065882 IC50 = 42900 nM T75570 CXC69T 137321158 IC50 = 384 nM T75570 CZOD53 137633880 IC50 = 189 nM T75570 C7BJY5 137636807 IC50 = 60 nM T75570 CO89DX 137649100 IC50 = 32 nM T75570 CINE03 137652514 IC50 = 266 nM T75570 C28QUP 137652864 IC50 = 57.3 nM T75570 CRWA29 139030520 IC50 > 10000 nM T75570 C2MD1Q 155513187 IC50 > 10000 nM T75570 C3NA2I 155519537 IC50 = 86 nM T75570 D03OKV 9844320 IC50 > 4.7 nM T75570 D06HVH 54613583 IC50 > 10000 nM T75570 D08RZB 11153014 IC50 = 2 nM T75570 D0C0ZC 11676786 IC50 = 51.2 nM T75570 D0CE3R 5312137 IC50 = 20 nM T75570 D0H1OK 11562302 IC50 = 10 nM T75570 D0N4LR 53469448 IC50 = 3195 nM T75570 D0O8AR 16097523 IC50 = 3 nM T75570 D0Y0BK 11524144 IC50 = 29.8 nM T79400 CGN48U 9827867 IC50 = 41 nM T79400 CW1G9B 10672666 IC50 > 10000 nM T79400 CW7Q2U 10895700 IC50 > 2500 nM T79400 CIQH43 11445130 IC50 = 3.4 nM T79400 C37MRI 16718808 IC50 = 12 nM T79400 CVO5L6 24748791 IC50 = 15 nM T79400 CS9TK6 38335241 IC50 > 200000 nM T79400 C25ELB 44143088 IC50 = 14454.4 nM T79400 CL0M7R 44143089 IC50 = 9772.37 nM T79400 C9QDC0 44143091 IC50 = 177827.94 nM T79400 C30CFX 44436704 IC50 = 40 nM T79400 CM83VP 72163524 IC50 > 10000 nM T79400 CWP85J 87360663 IC50 > 10000 nM T79400 CDCG19 122192781 Ki = 9 nM T79400 CD5SN7 122192782 Ki = 19.9 nM T79400 CJ6DA9 127028140 IC50 = 250 nM T79400 CD9KI3 127028141 IC50 = 80 nM T79400 C5MAS1 155510638 Ki = 0.13 nM T79400 CV8YT6 155516274 Ki = 1.8 nM T79400 CU80TM 155522954 Ki = 1.3 nM T79400 CU52QS 155545897 Ki = 1.6 nM T79400 CH2S6R 155546346 Ki = 0.44 nM T79400 CNZ1K5 155559920 Ki = 0.1 nM T79400 CTWE96 155561147 Ki = 0.3 nM T79400 D0Y5IQ 44255320 IC50 = 10000 nM T46937 D01BYB 5957 IC50 = 251188.64 nM T46937 D07VLY 31703 Ki > 10000 nM T46937 D09QBG 9854012 IC50 = 2 nM T46937 D0R3JB 4212 Ki > 10000 nM T46937 D0R6RC 54675777 Ki > 10000 nM T46937 D0WF7L 9871419 Ki = 1.995 nM T46937 D09VBE 16066663 IC50 < 10 nM T46937 D0KE4Z 5310954 EC50 = 1.3 nM T46937 D0UF2N 21706 IC50 < 250000 nM T46937 D0W4JI 11273179 IC50 = 16 nM T46937 D08NXX 5487281 EC50 = 20 nM T46937 D0M4LF 23649325 IC50 = 9 nM T46937 D0U7OU 3220 Ki > 10000 nM T46937 COE28J 7220 IC50 = 7430000 nM T46937 C4RT3E 10208 Ki > 10000 nM T46937 C73JPZ 10639 Ki > 10000 nM T46937 C9K3IP 78253 Ki = 17100 nM T46937 CFG7T8 80533 IC50 = 2060000 nM T46937 CZ8J9T 118348 Ki = 2390 nM T46937 CQ8JF0 131257 IC50 = 13000 nM T46937 C85EPW 167523 Ki = 2450 nM T46937 CKE6V0 196979 Ki > 10000 nM T46937 C1T2BC 442744 Ki > 10000 nM T46937 C20KPF 601138 IC50 = 1800000 nM T46937 C1VW6X 601157 IC50 = 1840000 nM T46937 C2JP7W 1149185 Ki = 4400 nM T46937 CHBV51 2741913 IC50 = 1260 nM T46937 CD68IW 2746549 IC50 = 320 nM T46937 C3KM2I 2746550 IC50 = 300 nM T46937 CX5MV4 4603056 IC50 = 1960000 nM T46937 CH8TP5 4742792 IC50 = 850 nM T46937 C7Z4OR 4742793 IC50 = 4000 nM T46937 C92LSY 4742794 IC50 = 3000 nM T46937 C7BQ1N 5492386 EC50 = 10 nM T46937 CW46EH 9823796 Ki = 2.512 nM T46937 C93YKA 9846875 Ki = 5.012 nM T46937 CPHL60 9850430 Ki = 5.012 nM T46937 CL73SJ 9866696 Ki > 10000 nM T46937 CEG2J4 9953334 Ki = 19.95 nM T46937 C5ZXR3 9969173 Ki = 660 nM T46937 C39LZS 9999105 EC50 = 40 nM T46937 CXQ0V1 10016898 EC50 = 24300 nM T46937 C4ST7G 10017729 EC50 = 66 nM T46937 C2F7DR 10098947 IC50 = 10800 nM T46937 CW2Q3B 10109037 Ki = 2990 nM T46937 CQRU04 10110666 IC50 > 2000 nM T46937 CV1I0S 10202847 Ki = 29 nM T46937 CT73IB 10260031 IC50 = 0.7 nM T46937 C61MTA 10292521 IC50 = 1800 nM T46937 CJ9W1G 10294407 IC50 = 690 nM T46937 C5COM0 10438063 IC50 = 316227.77 nM T46937 CMBN72 10480103 IC50 > 3000 nM T46937 CBQ9P2 10557443 IC50 = 0.7943 nM T46937 CI6FS2 11273178 IC50 = 16 nM T46937 C1TE6Z 11497605 IC50 = 690 nM T46937 CE6OM7 11503160 IC50 = 190 nM T46937 C2GL4P 11503687 IC50 = 190 nM T46937 C29GJZ 11504727 Ki = 19740 nM T46937 CDQ2L4 11504760 IC50 = 110 nM T46937 CHB3C7 11510273 Ki > 70000 nM T46937 C0EX1O 11519648 IC50 = 38 nM T46937 C2VW4K 11526078 IC50 = 90 nM T46937 CA7G1M 11532836 IC50 = 260 nM T46937 CT74ZJ 11560464 Ki > 70000 nM T46937 C7EWL5 11561528 IC50 = 180 nM T46937 C1V0UF 11561748 IC50 = 310 nM T46937 C2UH6Z 11569565 IC50 = 42 nM T46937 CG7D2T 11570029 IC50 = 210 nM T46937 CN62XG 11585280 Ki = 50.7 nM T46937 C03UQZ 11595497 IC50 = 40000 nM T46937 CUD1J5 11611428 Ki > 70000 nM T46937 CFZ48K 11620159 IC50 = 740 nM T46937 C0TDC2 11627317 IC50 = 560 nM T46937 CXM91P 11627571 IC50 = 250 nM T46937 CN3Z2G 11641496 IC50 = 650 nM T46937 C19DSA 11649277 Ki = 3130 nM T46937 C2IH1A 11656053 IC50 = 380 nM T46937 CI8VZ7 11663657 IC50 = 380 nM T46937 C1V2CG 11670815 Ki = 19 nM T46937 CH48LB 11677907 IC50 = 37 nM T46937 C85RIU 11684524 IC50 = 1100 nM T46937 C5IB0G 11684912 IC50 = 170 nM T46937 CPF5V6 11691323 IC50 = 370 nM T46937 CYK4J8 11697626 IC50 = 200 nM T46937 CKPR59 11699088 IC50 = 210 nM T46937 C3VW7P 11699570 IC50 = 800 nM T46937 C4P7MS 11706300 IC50 = 95 nM T46937 CA19OH 11706351 IC50 = 90 nM T46937 C15YHK 11712235 IC50 = 130 nM T46937 C9JTV2 11786496 IC50 = 11 nM T46937 CR9YO8 11950159 Ki = 8 nM T46937 C1OEX4 11950328 Ki = 172 nM T46937 CQ02OS 11950687 Ki = 3 nM T46937 C8PI6W 11955421 Ki = 35 nM T46937 C3WGI2 11955422 Ki = 397 nM T46937 CM07WK 11993787 IC50 = 250 nM T46937 CPS34X 12000684 IC50 = 97 nM T46937 CBW05G 12000767 IC50 = 142 nM T46937 CO94DG 12000848 IC50 = 266 nM T46937 CGV57W 12001028 IC50 = 428 nM T46937 CF0GO7 12001030 IC50 = 533 nM T46937 CRYI50 12001296 IC50 = 31 nM T46937 CTN8D0 12001479 IC50 = 73 nM T46937 CVLK47 12001567 IC50 = 53 nM T46937 C5UAK6 12001662 IC50 = 35 nM T46937 CWI0T3 12001755 IC50 = 21 nM T46937 C2AQN5 12002005 IC50 = 178 nM T46937 CXVM04 12002012 IC50 = 218 nM T46937 CH4S8D 14280990 EC50 = 1040 nM T46937 CD1Q4U 14280991 EC50 > 106000 nM T46937 C03ZNU 14280992 EC50 = 1910 nM T46937 CZ9WG1 14280994 EC50 > 106000 nM T46937 CL4AF3 14280995 EC50 > 100000 nM T46937 C1MK5R 14280996 EC50 = 1900 nM T46937 CCTP04 14280998 EC50 = 950 nM T46937 CXH95F 14280999 EC50 = 9110 nM T46937 CZ6N0W 14281000 EC50 = 280 nM T46937 CR1G8Y 14281001 EC50 = 20 nM T46937 C18OUM 14281003 EC50 = 420 nM T46937 CJ6VF1 14281004 EC50 = 180 nM T46937 CH1BM2 14281005 EC50 = 16 nM T46937 C9MY5X 14281006 EC50 = 0.7 nM T46937 CUCR03 14281008 EC50 = 60 nM T46937 CUFJ35 14281010 EC50 = 70 nM T46937 CQ8TE3 14281011 EC50 = 110 nM T46937 CSEC89 14281012 EC50 = 10860 nM T46937 CU0J8E 14281015 EC50 = 90 nM T46937 CDP92K 14281016 EC50 = 5 nM T46937 C6FCS9 14281018 EC50 = 50 nM T46937 CK3E1F 14281020 EC50 = 1400 nM T46937 CUDO17 14281023 EC50 = 150 nM T46937 CZ19AJ 14281024 EC50 = 140 nM T46937 CY8PC6 14281025 EC50 = 1 nM T46937 CBT8K9 14281026 EC50 = 1 nM T46937 C3F7MZ 14281027 EC50 = 250 nM T46937 C2CF9I 14281031 EC50 = 4840 nM T46937 CQ2YL0 14281033 EC50 = 770 nM T46937 CM1NW7 14281034 EC50 = 330 nM T46937 CEUF73 14281035 EC50 = 870 nM T46937 C7QJ4Y 14281036 EC50 = 50300 nM T46937 CWSR46 14281041 EC50 = 100 nM T46937 CZ1ML0 15005564 EC50 = 38 nM T46937 CTL89M 15005565 EC50 = 12 nM T46937 CRO7P1 15005566 EC50 = 360 nM T46937 CCO0S1 15005567 EC50 = 90 nM T46937 C74EYG 15005568 EC50 > 87500 nM T46937 C7RC1U 15005569 EC50 = 1660 nM T46937 CAC98D 15005570 EC50 = 9410 nM T46937 CW0UP4 15005571 EC50 = 3170 nM T46937 C6I0LA 15005572 EC50 = 520 nM T46937 CM63ZU 15005573 EC50 = 26700 nM T46937 CE0DR4 15005574 EC50 = 20 nM T46937 CAQ7J2 15005576 EC50 = 20 nM T46937 CTE39J 15005577 EC50 = 910 nM T46937 C8TQ6C 15005578 EC50 = 380 nM T46937 C5Z8QA 15005579 EC50 = 3020 nM T46937 CS17FZ 15005580 EC50 = 1330 nM T46937 CN13YK 15005581 EC50 = 190 nM T46937 CQ9Y7J 15005583 EC50 = 950 nM T46937 CJ72ZA 15005584 EC50 = 4 nM T46937 CVA9B0 15005585 EC50 = 55 nM T46937 C4PM2K 15005586 EC50 = 260 nM T46937 C95NSJ 15005588 EC50 = 180 nM T46937 CI60HD 15005590 EC50 = 6320 nM T46937 CDHV05 15005591 EC50 = 1320 nM T46937 C7VR0Q 15005592 EC50 = 5400 nM T46937 C7QZO0 15005594 EC50 = 390 nM T46937 C2V3LD 15005598 EC50 = 440 nM T46937 CPS49B 15005599 EC50 = 2690 nM T46937 CP6DI1 15005600 EC50 = 2470 nM T46937 C0Z6GL 15005601 EC50 = 2950 nM T46937 CTU06K 15005602 EC50 = 440 nM T46937 C23MUZ 15005603 EC50 = 430 nM T46937 CRA5G0 15005604 EC50 = 63100 nM T46937 C96YTU 15005605 EC50 = 210 nM T46937 CH7I9M 15005606 EC50 = 1070 nM T46937 CX9L6N 15005608 EC50 = 420 nM T46937 CYH3R2 15650856 IC50 = 41000 nM T46937 CU5TM4 15650857 IC50 = 47000 nM T46937 CZE1S0 15650858 IC50 = 44000 nM T46937 C36DUQ 15650859 IC50 = 58000 nM T46937 C43IYK 15650860 IC50 = 65000 nM T46937 C9R7HT 15650861 IC50 = 19000 nM T46937 COA37U 15650862 IC50 = 4000 nM T46937 C1TKE3 15650863 IC50 = 9000 nM T46937 CYF68T 15650864 IC50 = 43000 nM T46937 C3LJD1 15650865 IC50 = 12000 nM T46937 CCT4M2 15650866 IC50 = 2600 nM T46937 CE5J9H 15650867 IC50 = 43000 nM T46937 COA46R 15650868 IC50 = 7000 nM T46937 C9R8UL 15650869 IC50 = 14000 nM T46937 C93OLX 15650870 IC50 = 14000 nM T46937 C85VYP 15650871 IC50 = 5000 nM T46937 C7JUK0 15650872 IC50 = 4000 nM T46937 C8S5GB 15650873 IC50 = 4000 nM T46937 C07KVS 15650874 IC50 = 4300 nM T46937 C84LEG 15650875 IC50 = 3000 nM T46937 CGA45I 15650876 IC50 = 4000 nM T46937 CDF63H 15650877 IC50 = 11000 nM T46937 CIQ3E8 15650878 IC50 = 12000 nM T46937 C60ZLB 15650879 IC50 > 75000 nM T46937 CFUQ16 15650880 IC50 = 12000 nM T46937 C9KQ1O 15650881 IC50 = 2000 nM T46937 CKM82C 15650882 IC50 = 2800 nM T46937 CE2G8F 15650883 IC50 = 8000 nM T46937 CBHY29 15650884 IC50 > 75000 nM T46937 C5XCK6 15650885 IC50 > 75000 nM T46937 CAC01F 15650886 IC50 = 59000 nM T46937 C2OMY3 15650887 IC50 = 53000 nM T46937 C5ZF4J 15650888 IC50 = 41000 nM T46937 CBJ3X2 15650897 IC50 = 8900 nM T46937 CC8UZ0 15650898 IC50 = 69000 nM T46937 CLP60K 15650899 IC50 = 1400 nM T46937 CLF93J 15982392 IC50 = 88 nM T46937 C5U0ED 15982393 IC50 = 54 nM T46937 CUCB94 15983052 IC50 = 67 nM T46937 C7SN1C 15983053 IC50 = 10 nM T46937 C0KRQ7 15983055 IC50 = 290 nM T46937 CS97JR 15983175 IC50 = 12 nM T46937 CBOI12 15983301 IC50 = 79 nM T46937 C0O5BA 15983546 IC50 = 17 nM T46937 CNZ60E 15983670 IC50 = 32 nM T46937 C83NXU 15983672 IC50 = 2900 nM T46937 C8QR1T 16739091 IC50 = 210 nM T46937 CN3M1O 16739092 IC50 = 237 nM T46937 C5VMW8 16739093 IC50 = 36.2 nM T46937 CJ0B4K 16739094 IC50 = 41 nM T46937 CPXH49 16739123 IC50 = 53 nM T46937 C9YK5V 16739124 IC50 = 160 nM T46937 C3T8JD 16739125 IC50 = 211 nM T46937 CZXV43 16739157 IC50 = 13 nM T46937 C8YUX6 16739158 IC50 = 288 nM T46937 C8UT0S 18717762 Ki = 5.012 nM T46937 CIX18B 20300396 IC50 = 810000 nM T46937 C7I1XM 20638786 Ki = 79.43 nM T46937 C5R9GU 20690429 Ki = 1.585 nM T46937 CV5O1T 20690446 Ki = 0.2512 nM T46937 CFO0M2 22184796 IC50 = 890 nM T46937 C8VW6J 22184814 IC50 = 840 nM T46937 C3KYN9 22184858 IC50 = 520 nM T46937 CK39QS 22184864 IC50 > 3000 nM T46937 C2AG9D 22184925 IC50 = 1800 nM T46937 C2R1DL 22185065 IC50 = 1200 nM T46937 CP7R6Y 22185105 IC50 = 910 nM T46937 CIL9Z6 23642329 IC50 = 280 nM T46937 C7GV8K 23662455 Ki = 10000 nM T46937 C7P1SA 23662764 Ki > 10000 nM T46937 CYZK58 23664788 Ki = 12200 nM T46937 C67WBS 23672996 Ki > 10000 nM T46937 CN5OC4 23673110 Ki = 10000 nM T46937 CZ7SX0 23675739 Ki > 10000 nM T46937 C4HJO0 23718715 Ki > 10000 nM T46937 CHI5U8 24750557 IC50 = 83 nM T46937 CKSW41 24750561 IC50 = 580 nM T46937 C6ST2J 24750719 IC50 = 1900 nM T46937 CN5X0A 24750723 IC50 = 230 nM T46937 C42LRT 24750874 IC50 = 490 nM T46937 CBS78H 24750876 IC50 = 430 nM T46937 CF3TC8 24751017 IC50 = 2400 nM T46937 CH85JK 24751297 IC50 = 960 nM T46937 CWX59N 24751300 IC50 = 1100 nM T46937 C6JQ1Z 24751438 IC50 = 1200 nM T46937 CJB3P1 24751572 IC50 = 1800 nM T46937 C24TLB 24751574 IC50 = 920 nM T46937 CA8GF1 24751575 IC50 = 1100 nM T46937 CX7ZD3 24751576 IC50 = 450 nM T46937 CK9W7Z 24751577 IC50 = 700 nM T46937 CABO68 24751579 IC50 = 1600 nM T46937 C0KEY2 24751581 IC50 = 1700 nM T46937 CPJ35E 24751708 IC50 = 2000 nM T46937 C7YDT9 24751709 IC50 = 1100 nM T46937 CCO3F4 24751710 IC50 = 460 nM T46937 CY1GS7 24751711 IC50 = 960 nM T46937 C84SJB 24751712 IC50 = 380 nM T46937 CHC14Q 24751850 IC50 = 420 nM T46937 C8VPT2 24751851 IC50 = 600 nM T46937 CRZ2M3 24751995 IC50 = 2000 nM T46937 CV61HI 24751996 IC50 = 950 nM T46937 C57JFC 24751997 IC50 = 100 nM T46937 C8KLX7 24751998 IC50 = 600 nM T46937 CRO0A3 24751999 IC50 = 2600 nM T46937 CA03BZ 24752128 IC50 = 1000 nM T46937 CN82FY 24752129 IC50 = 1060 nM T46937 CSV5W3 24752130 IC50 = 180 nM T46937 C9RPZ4 24752131 IC50 = 190 nM T46937 CJ3R5H 24752269 IC50 = 1800 nM T46937 CV2HF0 24752270 IC50 = 350 nM T46937 C05FEI 24752271 IC50 = 500 nM T46937 C2O5VN 24752419 IC50 = 450 nM T46937 C10VIG 24752420 IC50 = 180 nM T46937 C96OHY 24752421 IC50 = 270 nM T46937 C2OX8U 24752422 IC50 = 320 nM T46937 C8RW1L 24752557 IC50 = 490 nM T46937 C0H7LB 24752558 IC50 = 1300 nM T46937 CZA1J9 24752559 IC50 = 950 nM T46937 C26MWN 24752560 IC50 = 1500 nM T46937 CDKW17 24752561 IC50 = 270 nM T46937 CLAN49 24752711 IC50 = 240 nM T46937 CK35PX 24786234 IC50 = 2 nM T46937 CXZ58T 24799317 IC50 = 23000 nM T46937 C4QT3E 24799834 IC50 = 45070 nM T46937 C3HA4N 24799835 IC50 = 57070 nM T46937 CMJA06 24801414 IC50 = 52 nM T46937 CZO0W8 24801416 IC50 = 11170 nM T46937 C68IKP 24801573 IC50 = 3110 nM T46937 CC86QR 24829442 Ki = 15 nM T46937 CICF42 24829780 Ki = 42 nM T46937 C5JQB6 24829943 Ki = 114 nM T46937 CLG45Z 24830601 Ki = 209 nM T46937 CHA2I6 24868313 Ki > 10000 nM T46937 CLBW37 24937181 Ki = 11 nM T46937 CAN92Q 24968874 IC50 = 16 nM T46937 C20GMW 25022501 IC50 = 243 nM T46937 CK85UZ 25165435 IC50 = 76 nM T46937 CQOU76 39073052 Ki = 2100 nM T46937 C3TS7K 44125995 Ki = 372 nM T46937 C2Z4BL 44126504 Ki > 5000 nM T46937 CHQO90 44128387 Ki = 283 nM T46937 C2GK9P 44128468 Ki = 42 nM T46937 C5X1AQ 44128900 Ki = 42 nM T46937 CTVG29 44128901 Ki = 23 nM T46937 CM3YG0 44128980 Ki = 30 nM T46937 C7DST0 44128981 Ki = 40 nM T46937 CMWY16 44128982 Ki = 193 nM T46937 C6X3YI 44128983 Ki = 82 nM T46937 CGC56I 44129058 Ki = 23 nM T46937 C85OKZ 44129060 Ki = 0.8 nM T46937 C52VAZ 44129136 Ki = 5 nM T46937 CPM7E0 44129137 Ki = 1.5 nM T46937 C8R6LJ 44129368 Ki = 105 nM T46937 COC12W 44129369 Ki = 7.7 nM T46937 C6VKN3 44129371 Ki = 71 nM T46937 C0Z4TY 44129445 Ki = 303 nM T46937 C3VR2G 44129446 Ki = 66 nM T46937 CK5SD1 44129447 Ki = 56 nM T46937 C7F2LI 44129448 Ki = 41 nM T46937 CGH08U 44129449 Ki = 33 nM T46937 CUH15M 44129451 Ki = 107 nM T46937 C5H3LE 44129522 Ki = 219 nM T46937 C47SDX 44129524 Ki = 27 nM T46937 CNM86R 44129525 Ki = 459 nM T46937 C5WP3I 44157464 Ki = 3760 nM T46937 CTZ81X 44157465 Ki = 884 nM T46937 C0LTK8 44157466 Ki = 10000 nM T46937 CJN39O 44157467 Ki > 10000 nM T46937 CJ4E6Y 44157518 Ki = 614 nM T46937 CI21HV 44157519 Ki = 63 nM T46937 CU5X8A 44157520 Ki = 541 nM T46937 CHF40V 44241562 IC50 = 8080 nM T46937 CL72TA 44295999 IC50 = 480 nM T46937 CH06ZN 44296001 IC50 = 2200 nM T46937 CJ7Z2M 44296486 IC50 = 170 nM T46937 CXZ0V1 44304081 IC50 = 35000 nM T46937 CTY4U2 44323790 EC50 = 960 nM T46937 C4D0ZF 44443917 IC50 = 100 nM T46937 CGP27V 44443919 IC50 = 0.3162 nM T46937 CLBC52 44443921 IC50 = 0.5012 nM T46937 CSN3M1 44443933 Ki = 3.162 nM T46937 CQR1P9 44443935 Ki = 1.995 nM T46937 CU3E5S 44443938 Ki = 5.012 nM T46937 C64HOJ 44443939 Ki = 0.631 nM T46937 CF7SB1 44452736 IC50 = 4730 nM T46937 CGI90J 44452737 IC50 = 1270 nM T46937 C9A8LW 44452878 IC50 = 616 nM T46937 CAT75E 44452879 IC50 = 1310 nM T46937 CR2M9J 44452898 IC50 = 40 nM T46937 C2IDA9 44452921 IC50 = 663 nM T46937 CJ08RK 44452925 IC50 = 2480 nM T46937 CK0E2B 44452926 IC50 = 2550 nM T46937 C96SQE 44452947 IC50 = 3800 nM T46937 C9LMZ4 44452951 IC50 = 2700 nM T46937 CK1AU7 44452952 IC50 = 580 nM T46937 CM60LZ 44452977 IC50 = 9900 nM T46937 C5XKP6 44452982 IC50 = 2490 nM T46937 CEW93M 44453009 IC50 = 4330 nM T46937 CM34EZ 44453032 IC50 = 495 nM T46937 C78BQV 44453107 IC50 = 201 nM T46937 CRS1M7 44453109 IC50 = 4860 nM T46937 C1DWQ9 44453110 IC50 = 2230 nM T46937 C0JN3W 44453131 IC50 = 2950 nM T46937 CJPF52 44453132 IC50 = 513 nM T46937 CEYV61 44456046 Ki = 1850 nM T46937 CA82XJ 44456077 Ki > 10000 nM T46937 C1DU4Z 44456078 Ki = 6760 nM T46937 C1W8IK 44456201 Ki = 10000 nM T46937 CL74DQ 44457247 IC50 = 8680 nM T46937 C6LWM3 44457249 IC50 = 3300 nM T46937 C56JUQ 44457251 IC50 = 522 nM T46937 CYB0H2 44457262 IC50 = 8290 nM T46937 CIP6B7 44457274 IC50 = 1820 nM T46937 C23NHF 44457276 IC50 = 16700 nM T46937 C9S6OQ 44457278 IC50 = 11710 nM T46937 C5Y2RW 44457290 IC50 = 27100 nM T46937 C0V3OU 44457292 IC50 = 4630 nM T46937 CD70CI 44457294 IC50 = 6540 nM T46937 CVT6W1 44457324 IC50 = 3060 nM T46937 C3D5SF 44457338 IC50 = 7590 nM T46937 C5ITD1 44457371 IC50 = 10690 nM T46937 CQI0O7 44457392 IC50 = 16880 nM T46937 C2UMA5 44457401 IC50 = 48 nM T46937 CTC7N5 44457411 IC50 = 12920 nM T46937 C6BAK3 44457422 IC50 = 23930 nM T46937 C78AUJ 44464779 IC50 = 3 nM T46937 C9XNT2 44554515 IC50 = 1 nM T46937 CTJQ59 44555026 IC50 = 100 nM T46937 C2OTX9 44583417 Ki > 10000 nM T46937 C2KWN7 44583454 Ki > 10000 nM T46937 C41BAQ 44583493 Ki = 25100 nM T46937 CD47MO 44583494 Ki = 10000 nM T46937 CVP5H0 44583549 Ki = 7070 nM T46937 CD5O7G 44583580 Ki = 1900 nM T46937 C9BM5G 44583581 Ki = 660 nM T46937 C4ZTQ0 44583637 Ki > 10000 nM T46937 CIA6S4 44608149 IC50 = 57 nM T46937 CW3XJ1 44610468 IC50 = 17 nM T46937 C3T6BG 44610518 IC50 = 270 nM T46937 CO7K2H 44610519 IC50 = 42 nM T46937 CG7RS8 44610522 IC50 = 130 nM T46937 CPQ09B 44610759 Ki = 5 nM T46937 C8BI6C 44610760 Ki = 4 nM T46937 CP68UD 44631970 Ki = 15 nM T46937 CIX15W 44631974 Ki = 2.1 nM T46937 C43HON 44762396 IC50 = 1540 nM T46937 C6K5ZT 45139236 Ki = 1.5 nM T46937 CYC57N 45139400 Ki = 69 nM T46937 C4TKJ3 45139401 Ki = 31 nM T46937 C9M7PY 45139402 Ki = 6.9 nM T46937 CGX5E1 45139403 Ki = 5.9 nM T46937 CR3ZA2 45139404 Ki = 10 nM T46937 CBR1T8 45139405 Ki = 1.3 nM T46937 CKJ3F7 45139406 Ki = 4.5 nM T46937 C23TQM 45139407 Ki = 12 nM T46937 CR48LE 45139408 Ki = 1.3 nM T46937 CV5Z1L 45139585 Ki = 11 nM T46937 CX0S1R 45139586 Ki = 6.9 nM T46937 CTA9Y2 45139587 Ki = 3.7 nM T46937 CN3F4K 45139588 Ki = 4.2 nM T46937 C9CB8Q 45139589 Ki = 5.3 nM T46937 C15JAY 45139590 Ki = 7.4 nM T46937 CDK5Q7 45139591 Ki = 7.5 nM T46937 CNL12Y 45139592 Ki = 10 nM T46937 CYJ3R6 45139764 Ki = 94 nM T46937 C2GTC1 45139765 Ki = 280 nM T46937 C4L8KR 45139766 Ki = 3.7 nM T46937 C6UQY5 45139767 Ki = 11 nM T46937 C96FBC 45139768 Ki = 3 nM T46937 CYF1Q0 45139769 Ki = 2.5 nM T46937 CR9T4K 45139770 Ki = 11 nM T46937 C38IDA 45139771 Ki = 2.4 nM T46937 C0Y5XP 45139772 Ki = 2.6 nM T46937 C0VN3U 45139773 Ki = 5.8 nM T46937 C5S8FZ 45139945 Ki = 18 nM T46937 CRQ05I 45139946 Ki = 79 nM T46937 CI9O6G 45139947 Ki = 47 nM T46937 CD9WJ2 45139948 Ki = 44 nM T46937 CU6V2B 45139949 Ki = 28 nM T46937 CAWB56 45139950 Ki = 3.7 nM T46937 CL09QD 45139951 Ki = 11 nM T46937 CDI3Y9 45139952 Ki = 7.9 nM T46937 CEC34T 45139953 Ki = 18 nM T46937 C96JYB 45139954 Ki = 8.8 nM T46937 C3PQS1 45139955 Ki = 13 nM T46937 CM7S2J 45139956 Ki = 7.9 nM T46937 C8BQ4F 45139957 Ki = 6.1 nM T46937 CQZ14O 45139958 Ki = 4.6 nM T46937 C9MWK0 45140154 Ki = 46 nM T46937 C6KZ5T 45140155 Ki = 15 nM T46937 C5H8ZC 45140156 Ki = 33 nM T46937 CZ5O9H 45140157 Ki = 42 nM T46937 CA3F2Q 45140158 Ki = 492 nM T46937 C7VG9C 45140159 Ki = 4.5 nM T46937 CJ5W6E 45140160 Ki = 20 nM T46937 CVY48K 45140161 Ki = 89 nM T46937 CH9ZS5 45140162 Ki = 18 nM T46937 CWL6A9 45140163 Ki = 8.6 nM T46937 C9RK4J 45140164 Ki = 11 nM T46937 C27UDM 45140165 Ki = 2.8 nM T46937 C32CMN 45140166 Ki = 4.4 nM T46937 CR2EO1 45140353 Ki = 196 nM T46937 C58XUB 45140361 Ki = 14 nM T46937 CSL0F1 45140362 Ki = 8.4 nM T46937 C1VGX4 45140363 Ki = 9.4 nM T46937 CUHA50 45140364 Ki = 4.5 nM T46937 CD4BF9 45140365 Ki = 2.6 nM T46937 CSM1K9 45140366 Ki = 3.2 nM T46937 C6PYZ9 45140367 Ki = 5.4 nM T46937 CHYK36 45140368 Ki = 5.8 nM T46937 C30VPY 45140551 Ki = 2 nM T46937 CUEF96 45140552 Ki = 1.5 nM T46937 CCPI40 45140553 Ki = 1.8 nM T46937 C0JX7Z 45140554 Ki = 1.7 nM T46937 C2PKQ0 45140555 Ki = 8.6 nM T46937 C9Z6RL 45140556 Ki = 3.8 nM T46937 CKZ19G 45140557 Ki = 3.6 nM T46937 C1A6PI 45140558 Ki = 2.8 nM T46937 C0A8CM 45140743 Ki = 45 nM T46937 CX2K5M 45140744 Ki = 45 nM T46937 CI1B0U 45140745 Ki = 112 nM T46937 C8P4YN 45140746 Ki = 39 nM T46937 CK53VS 45140748 Ki = 2.1 nM T46937 CFGH76 45140749 Ki = 5.5 nM T46937 CTH63Z 45140750 Ki = 45 nM T46937 CM32HO 45140751 Ki = 1.7 nM T46937 C45KFH 45140752 Ki = 8.4 nM T46937 CD5H9K 45140753 Ki = 8.3 nM T46937 C6WN2Z 45140754 Ki = 12 nM T46937 CA1PF4 45140927 Ki = 54 nM T46937 C8KI9O 45140928 Ki = 2.4 nM T46937 C9LEC4 45140929 Ki = 4 nM T46937 C76CDE 45140930 Ki = 3.3 nM T46937 CNB64P 45140931 Ki = 3.5 nM T46937 C9UT6B 45140932 Ki = 2.3 nM T46937 CF98ZN 45140933 Ki = 7.7 nM T46937 C7WH3A 45140934 Ki = 11 nM T46937 CL7RE6 45140935 Ki = 4.8 nM T46937 CB4A8S 45140936 Ki = 22 nM T46937 C4YBC2 45140937 Ki = 3.3 nM T46937 CN2E7I 45140938 Ki = 2.1 nM T46937 CH2AT1 45140939 Ki = 3.7 nM T46937 CPA02Z 45141128 Ki = 2.7 nM T46937 CYQM02 45141129 Ki = 5 nM T46937 CY7NU0 45141130 Ki = 64 nM T46937 C79QWL 45141131 Ki = 4 nM T46937 CF6TO0 45141133 Ki = 6 nM T46937 C7IVG1 45141134 Ki = 2.5 nM T46937 C8P3QC 45141135 Ki = 10 nM T46937 C8FN0X 45141136 Ki = 1 nM T46937 C7QN8R 45141341 Ki = 3.2 nM T46937 CSG1V2 45141342 Ki = 1.5 nM T46937 C3XIM0 45141343 Ki = 12 nM T46937 CBU59A 45141344 Ki = 5.7 nM T46937 CWQD34 45141345 Ki = 9.4 nM T46937 CC0P6E 45141347 Ki = 12 nM T46937 CK0PL3 45141578 Ki = 9.8 nM T46937 CVE0H2 45141579 Ki = 2.1 nM T46937 CQSN29 45141580 Ki = 5.5 nM T46937 CZ94QB 45141581 Ki = 15 nM T46937 C3S2PW 45141582 Ki = 20 nM T46937 C79LVU 45141583 Ki = 7.6 nM T46937 CAO1U8 45141584 Ki = 5 nM T46937 CTI7Y8 45141585 Ki = 7 nM T46937 CSCF14 45141770 Ki = 17 nM T46937 C8N6QH 45141771 Ki = 6.5 nM T46937 C2L0AO 45141772 Ki = 22 nM T46937 CP54ZM 45141773 Ki = 9 nM T46937 CZ06AP 45141774 Ki = 9.9 nM T46937 CDV5G3 45141776 Ki = 19 nM T46937 C94KUS 45141980 Ki = 10 nM T46937 CS81XD 45141981 Ki = 2.4 nM T46937 CG35EM 45141982 Ki = 22 nM T46937 C9Y8AH 45141983 Ki = 1.5 nM T46937 CK3S1X 45141984 Ki = 6.5 nM T46937 C2U6YC 45141985 Ki = 5.1 nM T46937 C5CQ9D 45141986 Ki = 2.5 nM T46937 C4IAD0 45141987 Ki = 4.5 nM T46937 CF6AD8 45142213 Ki > 5680 nM T46937 C6VG8P 45142216 Ki = 1.9 nM T46937 C47RYG 45142217 Ki = 1.1 nM T46937 CG98TA 45142218 Ki = 11 nM T46937 CAFL20 45142219 Ki = 3.3 nM T46937 C4LI9R 45142220 Ki = 5.3 nM T46937 C3TRE2 45142221 Ki = 3.9 nM T46937 CC7VE3 45142222 Ki = 10 nM T46937 CPSW54 45142223 Ki = 2.6 nM T46937 CH4N7O 45142445 Ki = 2.6 nM T46937 CM2DP3 45142446 Ki = 62 nM T46937 CYS85V 45142447 Ki = 94 nM T46937 CL5KF9 45142448 Ki = 120 nM T46937 C6E3XL 45142449 Ki = 68 nM T46937 C4STP8 45142450 Ki = 7.6 nM T46937 CFS9H3 45142451 Ki = 5.3 nM T46937 CFG74S 45142452 Ki = 5.3 nM T46937 CY43GD 45142453 Ki = 5.5 nM T46937 C6A7CG 45263658 Ki = 6.31 nM T46937 CGX80T 45267707 Ki = 1190 nM T46937 C86TKV 45267712 Ki > 5700 nM T46937 CJC9Q1 45267721 Ki = 7 nM T46937 CD1W5O 45267722 Ki = 96 nM T46937 C8GXD4 45267728 Ki = 92 nM T46937 C3AK2I 45267738 Ki = 157 nM T46937 C86BFJ 45267750 Ki = 49 nM T46937 C9NS3P 45267751 Ki = 12 nM T46937 CTK5Y2 45267776 Ki = 373 nM T46937 C2FD9O 45268593 Ki = 14 nM T46937 C5Q0YP 45268594 Ki = 28 nM T46937 CN4HX2 45268619 Ki = 26 nM T46937 C9B2IO 45268630 Ki = 31 nM T46937 C4U2CA 45268641 Ki = 93 nM T46937 CIB4K5 45268642 Ki = 15 nM T46937 CS0DF4 45268660 Ki > 5700 nM T46937 C7WJU9 45269438 Ki = 11 nM T46937 C9FA5L 45269454 Ki = 68 nM T46937 CU37SK 45269461 Ki = 23 nM T46937 CA6XK1 45269465 Ki = 270 nM T46937 CX4JK8 45269472 Ki = 20 nM T46937 CK3HU9 45269473 Ki = 95 nM T46937 CWNL09 45269482 Ki = 157 nM T46937 CV8F1O 45269483 Ki = 48 nM T46937 CS5GA3 45269484 Ki = 80 nM T46937 CR32NL 45269502 Ki > 5400 nM T46937 C2CEO3 45270266 Ki = 484 nM T46937 CI8QM6 45270267 Ki = 733 nM T46937 COWU62 45270274 Ki = 5.7 nM T46937 C41HAP 45270288 Ki = 328 nM T46937 CSEQ82 45270294 Ki = 214 nM T46937 C4A9PG 45270295 Ki = 81 nM T46937 CF0L5I 45270296 Ki = 35 nM T46937 CFZS57 45270300 Ki = 99 nM T46937 CSOT19 45270314 Ki = 39 nM T46937 CLEI08 45270318 Ki = 146 nM T46937 CPY1U9 45270321 Ki = 69 nM T46937 C34GWX 45270322 Ki = 47 nM T46937 C0HGU8 45270323 Ki = 10 nM T46937 CGBA08 45271082 Ki = 356 nM T46937 C8C4FS 45271092 Ki = 27 nM T46937 CV0P4Y 45271100 Ki = 43 nM T46937 C2SY0E 45271128 Ki = 190 nM T46937 C5Z7QD 45271145 Ki = 36 nM T46937 CK6C5N 45271154 Ki = 11 nM T46937 CPBF35 45271155 Ki = 18 nM T46937 CI0NU9 45271162 Ki = 15 nM T46937 C6XI2F 45271977 Ki = 1610 nM T46937 C7CHR1 45271978 Ki = 2440 nM T46937 CFN09J 45271984 Ki = 29 nM T46937 C41ZUD 45272035 Ki = 189 nM T46937 CYKJ35 45272036 Ki = 18 nM T46937 C3GQ2K 45272054 Ki = 40 nM T46937 CO4F1R 45272055 Ki = 34 nM T46937 CHV96U 45272074 Ki = 3640 nM T46937 C1M4YS 45272842 Ki = 455 nM T46937 C1RJ0T 45272846 Ki = 203 nM T46937 CE7WP6 45272861 Ki = 9.9 nM T46937 CM24LU 45272869 Ki = 3.5 nM T46937 C2RUJ8 45272880 Ki = 18 nM T46937 C9RUX5 45272881 Ki = 33 nM T46937 CYCS21 45272902 Ki = 209 nM T46937 CCDZ68 45273782 Ki = 76 nM T46937 CI1O0G 45273789 Ki = 64 nM T46937 CZRX73 45273798 Ki = 145 nM T46937 CZK63V 45273811 Ki = 99 nM T46937 C0HB9W 45273812 Ki = 35 nM T46937 CF92SN 45273818 Ki = 24 nM T46937 C8D0IE 45273819 Ki = 14 nM T46937 C21EFP 45273820 Ki = 7 nM T46937 C5SAO6 45485848 Ki = 12 nM T46937 CO4N6X 45485849 Ki = 1.2 nM T46937 C9A1QE 45485850 Ki = 1.2 nM T46937 CA52GP 45485851 Ki = 55 nM T46937 C7SEY6 45485852 Ki = 72 nM T46937 CW9ZK8 45485853 Ki = 27 nM T46937 CW56DP 45485854 Ki = 184 nM T46937 CVO1I8 45485855 Ki = 2.8 nM T46937 C57UAI 45485856 Ki = 11 nM T46937 C9XPS3 45485857 Ki = 19 nM T46937 CJ35NO 45485858 Ki = 16 nM T46937 CF15OM 45485859 Ki = 2.2 nM T46937 C30RBF 45485860 Ki = 31 nM T46937 C0O9SQ 45485861 Ki = 15 nM T46937 CQL67G 45485862 Ki = 5.7 nM T46937 CP1F0U 45485863 Ki = 12 nM T46937 C9F8JX 45485864 Ki = 123 nM T46937 CD4ZJ1 45485865 Ki = 42 nM T46937 CI8O1H 45485880 Ki = 4.5 nM T46937 CP0YJ1 45485881 Ki = 22 nM T46937 C3Q7DF 45485882 Ki = 17 nM T46937 CD5N2R 45485883 Ki = 70 nM T46937 CI2Y7S 45485884 Ki = 1.2 nM T46937 CX0NC7 45485885 Ki = 5.2 nM T46937 CWK64B 45485886 Ki = 1 nM T46937 C6Q5RW 45485887 Ki = 11 nM T46937 CJU65A 45485888 Ki = 2.5 nM T46937 CN0S5H 45485889 Ki = 1.2 nM T46937 C26XAU 45485890 Ki = 4.8 nM T46937 CL7EW0 45485891 Ki = 38 nM T46937 CZ2V1S 45485892 Ki = 4.1 nM T46937 CN5ZT0 45485893 Ki = 19 nM T46937 C4PE7J 45485894 Ki = 9.4 nM T46937 CXP98J 45485895 Ki = 35 nM T46937 C9D6YA 45485896 Ki = 2.7 nM T46937 C2WC1A 45485897 Ki = 11 nM T46937 CET6H3 45485898 Ki = 0.69 nM T46937 CP1NK2 45485899 Ki = 8.4 nM T46937 C4NS9G 45485900 Ki = 2 nM T46937 CL52BA 45485901 Ki = 22 nM T46937 C1AG4M 45485902 Ki = 3.7 nM T46937 CT8FO2 45485903 Ki = 29 nM T46937 CW78YS 45485904 Ki = 1.2 nM T46937 CC83HT 45485905 Ki = 5.8 nM T46937 C7K4OZ 45485906 Ki = 2.9 nM T46937 C8COX6 45485907 Ki = 14 nM T46937 CS1PN6 45485908 Ki = 2.6 nM T46937 CDLE53 45485909 Ki = 6.8 nM T46937 CG3W8L 45485910 Ki = 2.1 nM T46937 CT6ZU5 45485911 Ki = 2.3 nM T46937 CZW7Y2 45485912 Ki = 12 nM T46937 CR1YJ9 45485913 Ki = 7.5 nM T46937 CM26UH 45485914 Ki = 1.7 nM T46937 CR76LO 45485915 Ki = 1.5 nM T46937 C5NA1E 45485916 Ki = 7.4 nM T46937 C7HP0T 45485917 Ki = 1.3 nM T46937 CMO8T0 45485918 Ki = 2.9 nM T46937 CY34QO 45485919 Ki = 5.9 nM T46937 CNZ61J 45485920 Ki = 3 nM T46937 CA4RQ5 45485921 Ki = 9.4 nM T46937 C5H9DG 45485922 Ki = 1.2 nM T46937 C8IG5O 45485928 Ki = 11 nM T46937 CYM5B3 45485929 Ki = 2.2 nM T46937 CIWL84 45485930 Ki = 11 nM T46937 CEY93C 45485931 Ki = 0.61 nM T46937 C46HGC 45485932 Ki = 0.4 nM T46937 CRUQ16 45485933 Ki = 2.7 nM T46937 CK0S4N 45485934 Ki = 3 nM T46937 CH8ZV1 45485935 Ki = 2.8 nM T46937 C9H2MB 45485936 Ki = 2.1 nM T46937 C9AZ1U 45485937 Ki = 4.2 nM T46937 CT5P0G 45485938 Ki = 1.4 nM T46937 C7CP1G 45485939 Ki = 5 nM T46937 CNJP56 45485940 Ki = 7.4 nM T46937 CV9G4L 45485941 Ki = 5.3 nM T46937 CC57DL 45485942 Ki = 7.1 nM T46937 C2EQO3 45485943 Ki = 0.71 nM T46937 CPA16Y 45485944 Ki = 10 nM T46937 CME01Q 45485945 Ki = 8.4 nM T46937 CCZ16M 45485946 Ki = 12 nM T46937 COXP14 45485947 Ki = 4.3 nM T46937 C15VLC 45485948 Ki = 8.1 nM T46937 CQ17ES 45485949 Ki = 2 nM T46937 CB3C4P 45485950 Ki = 10.2 nM T46937 C1T4GP 45485951 Ki = 8.4 nM T46937 CLVB13 45485952 Ki = 0.99 nM T46937 CZ6W9U 45485953 Ki = 2 nM T46937 CRNG05 45485954 Ki = 3.5 nM T46937 C0G7VB 45485955 Ki = 1.3 nM T46937 C0H7QZ 45485956 Ki = 2.5 nM T46937 C73WXS 45485957 Ki = 0.38 nM T46937 C1MG8V 45485958 Ki = 0.6 nM T46937 C7F9WV 45485959 Ki = 0.79 nM T46937 C2DFB9 45485960 Ki = 3.6 nM T46937 CMQ15J 45485961 Ki = 0.83 nM T46937 C9IA7C 45485962 Ki = 0.7 nM T46937 CJ53NZ 45485963 Ki = 0.46 nM T46937 CF72IM 45485964 Ki = 3.6 nM T46937 CP0S1Q 45485965 Ki = 0.9 nM T46937 C5OIB6 45485966 Ki = 0.67 nM T46937 CM59YQ 45485967 Ki = 3.1 nM T46937 CU9M0E 45485968 Ki = 0.92 nM T46937 CQE2D6 45485969 Ki = 1.6 nM T46937 CQWH31 45487789 Ki = 223 nM T46937 CU12YR 45487790 Ki = 213 nM T46937 C93PEY 45487796 Ki = 130 nM T46937 CGAY47 45487800 Ki = 36 nM T46937 C6BJ1X 45487801 Ki = 539 nM T46937 C1C6BE 45487809 Ki = 37 nM T46937 CUTP63 45487813 Ki = 191 nM T46937 CA53DG 45487817 Ki = 27 nM T46937 CN17LS 45487821 Ki = 68 nM T46937 C7TO3S 45487837 Ki = 240 nM T46937 CO68ZR 45487838 Ki = 839 nM T46937 CR24MB 45487841 Ki = 37 nM T46937 CKG8Z5 45487842 Ki = 78 nM T46937 CIOH61 45487843 Ki = 295 nM T46937 C47CSK 45487844 Ki = 380 nM T46937 C19MHZ 45487850 Ki = 31 nM T46937 COCJ34 46232830 Ki = 3.8 nM T46937 CQP62R 46232879 Ki = 1.5 nM T46937 CWA82V 46232880 Ki = 7.5 nM T46937 CKN5C7 46232881 Ki = 4 nM T46937 C09PJV 46232882 Ki = 11 nM T46937 CI8Y4W 46232883 Ki = 2.8 nM T46937 CJ0W1O 46232884 Ki = 12 nM T46937 C9KY1C 46232885 Ki = 8 nM T46937 C0Z2DI 46232886 Ki = 25 nM T46937 CV9PC5 46232887 Ki = 0.79 nM T46937 CC20BA 46232888 Ki = 6.5 nM T46937 C9W8XE 46232889 Ki = 7.9 nM T46937 C6DS2Y 46232890 Ki = 0.58 nM T46937 C1SK2F 46232891 Ki = 4.3 nM T46937 C7A1BX 46232892 Ki = 6 nM T46937 CB2SN5 46232893 Ki = 2.6 nM T46937 CL21DR 46232894 Ki = 0.98 nM T46937 CKZS79 46232895 Ki = 12 nM T46937 CR5CV6 46232896 Ki = 1.1 nM T46937 CPJ41D 46232897 Ki = 4 nM T46937 CXM05D 46232898 Ki = 4.8 nM T46937 C8CMR5 46232899 Ki = 1.2 nM T46937 C8RP5H 46232900 Ki = 2.8 nM T46937 C4M9TH 46232901 Ki = 6.5 nM T46937 CT3CB2 46232902 Ki = 15 nM T46937 CM4S2A 46232903 Ki = 29 nM T46937 CVW47M 46232904 Ki = 13 nM T46937 CW5C6S 46232905 Ki = 8.3 nM T46937 CT1V2F 46232906 Ki = 6.3 nM T46937 CT0JF6 46232907 Ki = 4.5 nM T46937 CM4FR7 46232908 Ki = 8.5 nM T46937 CCA21B 46232909 Ki = 8.4 nM T46937 C2LX4J 46232910 Ki = 8.9 nM T46937 CL6KU2 46232911 Ki = 1.7 nM T46937 C9N2DT 46232912 Ki = 4.9 nM T46937 C3EWR0 46232913 Ki = 5.9 nM T46937 C4Q7ED 46232914 Ki = 5.2 nM T46937 CSX0C1 46232915 Ki = 22 nM T46937 C5V7ZC 46232916 Ki = 16 nM T46937 C5K0AF 46232917 Ki = 2.8 nM T46937 CG2Q0P 46232918 Ki = 6.3 nM T46937 C2CBX6 46232919 Ki = 5.9 nM T46937 CP4DL3 46232920 Ki = 12 nM T46937 CWE0H5 46232921 Ki = 10 nM T46937 C6OJ8N 46232922 Ki = 18 nM T46937 C2M9NJ 46232923 Ki = 16 nM T46937 C96VNX 46232924 Ki = 31 nM T46937 CR6W5O 46232925 Ki = 22 nM T46937 CT21LP 46232926 Ki = 5.5 nM T46937 C9F3OL 46232927 Ki = 11 nM T46937 CQ5IB9 46232928 Ki = 7.3 nM T46937 C9FUS3 46232929 Ki = 9.9 nM T46937 CK4T7U 46232930 Ki = 10 nM T46937 CF18EQ 46232931 Ki = 17 nM T46937 C04DRM 46232932 Ki = 26 nM T46937 CXT3Q5 46232933 Ki = 13 nM T46937 C2HJ0E 46232934 Ki = 5 nM T46937 C1O5RS 46232935 Ki = 3.5 nM T46937 CW5F1D 46232936 Ki = 21 nM T46937 CE3R8K 46232937 Ki = 31 nM T46937 CTB0W6 46232940 Ki = 1.7 nM T46937 CNV89R 46232941 Ki = 2.6 nM T46937 CS60LF 46232942 Ki = 1.7 nM T46937 CB3T7O 46232943 Ki = 1.4 nM T46937 C7DO0E 46232944 Ki = 2.5 nM T46937 CYW60D 46232945 Ki = 2 nM T46937 C3U5NH 46232946 Ki = 5.5 nM T46937 C8XGB6 46232947 Ki = 3.3 nM T46937 CO0P1Y 46232948 Ki = 7.1 nM T46937 CNOI84 46232949 Ki = 0.64 nM T46937 CX1C6B 46232950 Ki = 1.7 nM T46937 CV82XQ 46232951 Ki = 2 nM T46937 CIC1X6 46233093 Ki > 3590 nM T46937 CCA2D3 46233094 Ki > 3590 nM T46937 CNRH34 46233095 Ki = 842 nM T46937 C8H1KS 46233096 Ki = 288 nM T46937 CIX16N 46233130 Ki = 277 nM T46937 CT7IR5 46233131 Ki = 613 nM T46937 C14FKB 46233132 Ki = 55 nM T46937 CRPZ16 46233133 Ki = 54 nM T46937 CZ42KE 46233134 Ki = 842 nM T46937 CBT14W 46233174 Ki = 9 nM T46937 C2RIO9 46233175 Ki = 42 nM T46937 CM01FC 46233176 Ki = 8 nM T46937 CT56IZ 46233222 Ki = 132 nM T46937 C24DJR 46233223 Ki = 4.9 nM T46937 CQ9G7I 46233224 Ki = 6 nM T46937 C1C5YP 46233225 Ki = 6.2 nM T46937 CYG90O 46233226 Ki = 9.1 nM T46937 C3A5QP 46233227 Ki = 8.5 nM T46937 C0UVF8 46233228 Ki = 3 nM T46937 CWIN59 46233229 Ki = 2.3 nM T46937 C5Y9MB 46233230 Ki = 25 nM T46937 CVLW59 46233231 Ki = 5.7 nM T46937 C3UP9V 46233232 Ki = 4.1 nM T46937 C2VES7 46233233 Ki = 2.7 nM T46937 CH1V0B 46233234 Ki = 1.4 nM T46937 CD8K6M 46233235 Ki = 4.7 nM T46937 C2LZ8X 46233236 Ki = 5.8 nM T46937 C05LBX 46233237 Ki = 3.2 nM T46937 CYA83J 46233238 Ki = 9.2 nM T46937 C5ZGP7 46233239 Ki = 43 nM T46937 C57LNR 46233240 Ki = 11 nM T46937 CFLO71 46233241 Ki = 1.4 nM T46937 CBT2O9 46233242 Ki = 1.9 nM T46937 C26MHU 46233243 Ki = 1.7 nM T46937 C0NK3C 46233290 Ki > 5400 nM T46937 CX8Y9L 46233321 Ki > 5700 nM T46937 CJG70T 46233322 Ki = 373 nM T46937 C6IG4P 46233323 Ki = 3640 nM T46937 CXE56T 46233324 Ki = 28 nM T46937 CXEF72 46233325 Ki = 1.5 nM T46937 C2MK7D 46233326 Ki = 4.9 nM T46937 C3ZCA6 46233327 Ki = 2.8 nM T46937 C35TNK 46233328 Ki = 3.6 nM T46937 CD92SU 46233329 Ki = 2.4 nM T46937 CL5SQ7 46233330 Ki = 11 nM T46937 C8MH6O 46233354 Ki = 484 nM T46937 C0E7KD 46233355 IC50 = 64 nM T46937 C48ZWF 46233356 Ki = 1190 nM T46937 C8BG5H 46233357 Ki = 733 nM T46937 CD0JE2 46233386 Ki = 1610 nM T46937 CHR32N 46233387 Ki > 5700 nM T46937 C49FAM 46233388 Ki = 1430 nM T46937 C86YOM 46233389 Ki = 1310 nM T46937 CWO5Q7 46233451 Ki = 87 nM T46937 C0IAC3 46233532 Ki > 3800 nM T46937 CU27WP 46233553 Ki > 3800 nM T46937 C8N0DY 46233554 Ki > 3590 nM T46937 C8W6EH 46233555 Ki > 2710 nM T46937 C5C6IN 46233586 Ki > 3590 nM T46937 CVT9H3 46233587 Ki > 3590 nM T46937 C69VFP 46233588 Ki > 3590 nM T46937 CO52XP 46233589 Ki = 3100 nM T46937 CKP38S 46233630 Ki = 1430 nM T46937 CXE6J5 46233631 Ki > 3590 nM T46937 C0Q9JC 46233632 Ki > 3590 nM T46937 C6P7IQ 46233668 Ki = 1880 nM T46937 C7QIO4 46233669 Ki > 3590 nM T46937 C5BMY9 46233670 Ki > 3590 nM T46937 CQNZ48 46241018 IC50 = 1400 nM T46937 CVP5D0 46241232 IC50 = 310 nM T46937 CEB52S 51032397 IC50 = 820000 nM T46937 CD9C1M 53233471 IC50 = 110 nM T46937 CR98BF 53350233 IC50 > 20000 nM T46937 CZI4D6 54579992 IC50 > 33000 nM T46937 C37EUW 54579993 IC50 > 33000 nM T46937 COH9F8 54579994 IC50 > 33000 nM T46937 CC4H9D 54579995 IC50 = 5500 nM T46937 CA95EC 54579996 IC50 = 3000 nM T46937 CA9W6B 54579997 IC50 = 4600 nM T46937 CD6R5X 54580043 IC50 > 33000 nM T46937 C2R4NO 54580044 IC50 = 29000 nM T46937 C01JXK 54580185 IC50 = 8500 nM T46937 C97ZBQ 54580993 IC50 = 2700 nM T46937 C4XDL0 54580994 IC50 = 9600 nM T46937 CT8S3D 54580995 IC50 = 2700 nM T46937 CI3A4F 54581027 IC50 = 760 nM T46937 CE4O3T 54581187 IC50 > 33000 nM T46937 C5H8MZ 54582036 IC50 > 33000 nM T46937 CO0AU9 54582209 IC50 > 33000 nM T46937 C4WH5A 54583010 IC50 > 33000 nM T46937 CPG8J3 54583974 IC50 = 4600 nM T46937 CSW27C 54583975 IC50 = 3000 nM T46937 C0B6QV 54584163 IC50 = 3800 nM T46937 CSM50F 54584960 IC50 = 2100 nM T46937 CS0YL3 54585098 IC50 = 8600 nM T46937 CDKR61 54585884 IC50 > 33000 nM T46937 CC8WI6 54585885 IC50 = 1800 nM T46937 CMIX30 54586076 IC50 = 890 nM T46937 CAB1F6 54732982 IC50 = 35000 nM T46937 C6MGO8 59534139 IC50 = 3 nM T46937 CTJM21 59534140 IC50 = 16 nM T46937 C8Z5FQ 60150614 IC50 > 10000 nM T46937 CA1KI7 66575818 IC50 = 1800 nM T46937 CM5CX3 66575819 IC50 = 5.1 nM T46937 C9EUN4 66575821 IC50 = 275 nM T46937 CFBA98 66575899 IC50 = 17 nM T46937 CC8K0B 66576220 IC50 = 7 nM T46937 CWD98Y 66576221 IC50 = 48 nM T46937 CXF02Q 66576296 IC50 = 15 nM T46937 C3JR2F 66576297 IC50 = 20 nM T46937 CU8A4R 66576298 IC50 = 27 nM T46937 CGRD93 66576377 IC50 = 22 nM T46937 C7EHJ6 66576448 IC50 = 500 nM T46937 CM8T2U 66576450 IC50 = 26 nM T46937 CXEP01 66576451 IC50 = 48 nM T46937 CA48WV 66576530 IC50 = 11 nM T46937 CLE6I7 66576610 IC50 = 50 nM T46937 CDH3K2 66854409 Ki = 613 nM T46937 C1NXY6 66854417 Ki = 238 nM T46937 C4EZJ9 66854424 Ki = 56 nM T46937 CK0MP7 66854575 Ki = 130 nM T46937 CW08UL 66854714 Ki = 183 nM T46937 CIM37J 66854759 Ki = 6.5 nM T46937 C04PRO 66854841 Ki = 5.7 nM T46937 C3J2VK 66854919 Ki = 180 nM T46937 CJY0F5 66855084 Ki = 56 nM T46937 CL65PY 66855175 Ki = 111 nM T46937 CBRU59 66855176 Ki > 5000 nM T46937 C9BKL3 66855197 Ki = 20 nM T46937 CS8B3V 66855285 Ki = 22 nM T46937 CR6B2X 66855732 Ki = 3.1 nM T46937 CR7W0Y 66855824 Ki = 7.3 nM T46937 CF0EX4 66855902 Ki = 5 nM T46937 CEJ1Z9 66855932 Ki = 48 nM T46937 CC4FR1 66856100 Ki = 172 nM T46937 C9E5DR 66856658 Ki = 51 nM T46937 CE45CN 66856790 Ki = 54 nM T46937 C4Z5AD 66856844 Ki = 19 nM T46937 CT16XL 66856952 Ki = 202 nM T46937 CIA84K 66856999 Ki = 207 nM T46937 C5AT4J 66857005 Ki = 80 nM T46937 CON4R7 66919940 Ki = 242 nM T46937 C1MNH8 66919958 Ki = 2720 nM T46937 CG0Y7J 66919996 Ki = 249 nM T46937 C3P4ZO 66920261 Ki = 574 nM T46937 CR1J5S 67459247 IC50 = 46 nM T46937 CB29XL 67459391 IC50 = 198 nM T46937 C0UXC9 67459556 IC50 = 95.5 nM T46937 C7NWK1 67459575 IC50 = 27 nM T46937 CPKE56 67460268 IC50 = 25 nM T46937 C2PYM3 67460312 IC50 = 100 nM T46937 CSA0H7 67460401 IC50 = 169 nM T46937 C63EOD 67460624 IC50 = 11 nM T46937 C3NWK7 67460741 IC50 = 129 nM T46937 CEHN20 67460935 IC50 = 36 nM T46937 C2KJ5P 67460979 IC50 = 52 nM T46937 CFDP23 67461519 IC50 = 257 nM T46937 CL5Q6D 67461716 IC50 = 21 nM T46937 CGBJ01 67461890 IC50 = 279 nM T46937 CA4E9H 67462098 IC50 = 40 nM T46937 CIXA56 67462183 IC50 = 56 nM T46937 CBHW91 67462328 IC50 = 201 nM T46937 C8W6XY 67462688 IC50 = 177 nM T46937 CMH1P6 67462816 IC50 = 59.5 nM T46937 CU90BR 67463039 IC50 = 122 nM T46937 CJD0F6 67463112 IC50 = 162 nM T46937 C6YF1M 67463220 IC50 = 52 nM T46937 CN0C3L 67463698 IC50 = 223 nM T46937 CRU26C 67463976 IC50 = 98 nM T46937 C5E4VR 67464143 IC50 = 2780 nM T46937 C6IO7J 67464394 IC50 = 219 nM T46937 CF59TE 68529945 Ki > 70000 nM T46937 C4VFI2 68530100 Ki > 70000 nM T46937 CNR0K9 68556549 IC50 = 190 nM T46937 CE7G0I 68556579 IC50 = 11000 nM T46937 CBP40H 68842714 IC50 = 680 nM T46937 C6TUH7 68910943 IC50 = 59 nM T46937 CDAK52 68911008 IC50 = 3200 nM T46937 C4VN1H 68911027 IC50 = 240 nM T46937 CV5HD9 68911088 IC50 = 110 nM T46937 CQC63W 68911120 IC50 = 710 nM T46937 CMQS54 68911155 IC50 = 27 nM T46937 CYAK78 68911205 IC50 = 39 nM T46937 C8QND7 68911289 IC50 = 9.5 nM T46937 C1B4XM 68913141 IC50 = 86 nM T46937 C87OTJ 68913220 IC50 = 690 nM T46937 CN61KV 68913927 IC50 = 190 nM T46937 C89ZLC 68914580 IC50 = 380 nM T46937 CE6OV1 68916097 IC50 = 3800 nM T46937 C70RGD 68916926 IC50 = 22 nM T46937 CP1NH0 68918061 IC50 = 240 nM T46937 CO43WI 69223141 IC50 = 220 nM T46937 C02UFD 69224054 IC50 = 7 nM T46937 C7SQT4 69224555 IC50 = 6 nM T46937 CCV7T0 69224603 IC50 = 180 nM T46937 C7Z9LF 69224988 IC50 = 30 nM T46937 C6EUY5 70618043 IC50 = 1070000 nM T46937 CI23ZK 70683418 Ki = 24 nM T46937 CKX7O8 70687668 Ki = 26 nM T46937 C84IOJ 70922234 IC50 = 46 nM T46937 CG56TS 71449929 Ki = 536 nM T46937 CGJ70Y 71455298 Ki = 173 nM T46937 C3LB1G 71462475 Ki = 958 nM T46937 CQ1SO4 71462476 Ki > 5000 nM T46937 CU8LY5 71607553 IC50 = 1730 nM T46937 CC4Y0J 71607589 IC50 = 280 nM T46937 CAH29B 71607592 IC50 = 16300 nM T46937 CI4PG7 71607631 IC50 = 220 nM T46937 CB3ED0 71607632 IC50 = 350 nM T46937 CTJ57B 71607634 IC50 = 11280 nM T46937 C0M4ED 71607663 IC50 = 6350 nM T46937 C6SLH7 71607664 IC50 = 1670 nM T46937 CJ3O6U 71607665 IC50 = 4820 nM T46937 CI04FH 71607666 IC50 = 1970 nM T46937 C4G8TJ 71607689 IC50 = 330 nM T46937 CRD4I9 71625797 Ki > 30000 nM T46937 CR0HK1 71740352 IC50 = 3700 nM T46937 CD8HZ2 71740353 IC50 = 5300 nM T46937 C8YZ2K 71740354 IC50 > 33000 nM T46937 CD6QV9 71740705 IC50 = 9300 nM T46937 C3UA0H 71740819 IC50 = 660 nM T46937 C9A2RG 73294137 IC50 = 230 nM T46937 CWV9G3 73603967 IC50 = 7 nM T46937 CT0FK7 74220534 IC50 = 40 nM T46937 C4IC1L 85909513 IC50 = 1300000 nM T46937 CUA2D5 85909522 IC50 = 1050000 nM T46937 CES8C1 90078535 IC50 > 10000 nM T46937 CCEV76 90644279 IC50 = 270 nM T46937 C1DML0 90644280 IC50 = 11500 nM T46937 C8E0CO 90644281 IC50 = 93 nM T46937 CXZ8K5 90644282 IC50 = 20000 nM T46937 C27IDK 118710241 IC50 = 46 nM T46937 CZ1D6E 118710242 IC50 = 76 nM T46937 C6JY4L 118710243 IC50 = 291 nM T46937 C2K0BX 118710244 IC50 = 23 nM T46937 C6HN8Y 118710245 IC50 = 39 nM T46937 CSAX95 118710246 IC50 = 43 nM T46937 C3PM1C 118710247 IC50 = 9 nM T46937 C10PNU 118711064 IC50 = 15000 nM T46937 CQGB17 118711065 IC50 = 272 nM T46937 CH28LI 118711066 IC50 = 93 nM T46937 CZAC38 118711067 IC50 = 800 nM T46937 CX24WK 118711069 IC50 = 31 nM T46937 C8KD4V 118711070 IC50 = 61 nM T46937 CA9VN3 118711071 IC50 = 94 nM T46937 CWD74Q 118711072 IC50 = 92 nM T46937 CGH0Q5 118711073 IC50 = 194 nM T46937 C9BG2N 118711074 IC50 = 124 nM T46937 CB08DC 118711075 IC50 = 61 nM T46937 C0FOK2 118711076 IC50 = 88 nM T46937 CP9DZ6 118711077 IC50 = 139 nM T46937 C5QB8J 118711078 IC50 = 47 nM T46937 CQZ27P 118711079 IC50 = 71 nM T46937 CE16LZ 118711080 IC50 = 84 nM T46937 C21ZCF 118711081 IC50 = 95 nM T46937 C7EXA6 118711082 IC50 = 71 nM T46937 CV6LC1 118711083 IC50 = 115 nM T46937 CT52KG 118711084 IC50 = 94 nM T46937 C7QFM6 118711085 IC50 = 87 nM T46937 C9CPJ3 118711086 IC50 = 46 nM T46937 C4QI0G 118711087 IC50 = 65 nM T46937 CC4NM8 118711088 IC50 = 73 nM T46937 C7S5GQ 118711089 IC50 = 111 nM T46937 C9VB0Y 118711090 IC50 = 100 nM T46937 CQC05Z 118711091 IC50 = 117 nM T46937 C9BZ8T 118711092 IC50 = 89 nM T46937 CCS8T0 118711093 IC50 = 106 nM T46937 C63SGU 118711094 IC50 = 33 nM T46937 C2TRX6 118711095 IC50 = 66 nM T46937 CH5X7F 118711096 IC50 = 121 nM T46937 CH2ST8 118711097 IC50 = 41 nM T46937 C1YR4C 118711098 IC50 = 29 nM T46937 CV7S2E 118711099 IC50 = 44 nM T46937 CN2T0A 118711100 IC50 = 76 nM T46937 C4FPM5 118711101 IC50 = 82 nM T46937 C8EP3X 118711102 IC50 = 27 nM T46937 CH42SK 118711172 IC50 = 102 nM T46937 CVI36F 118711173 IC50 = 28 nM T46937 CI94EL 118711174 IC50 = 19 nM T46937 CK78YV 118711175 IC50 = 19 nM T46937 C7B0TZ 118711176 IC50 = 66 nM T46937 C28QNW 118711177 IC50 = 15 nM T46937 C41DUA 118711178 IC50 = 86 nM T46937 CHV13J 118711179 IC50 = 70 nM T46937 C93IST 118711180 IC50 = 12 nM T46937 CW0NK6 118711181 IC50 = 48 nM T46937 CV02RP 118711182 IC50 = 34 nM T46937 C9QY3L 118711183 IC50 = 76 nM T46937 C63OXP 118711184 IC50 = 118 nM T46937 C64VUZ 118711185 IC50 = 138 nM T46937 C5NW9I 118711186 IC50 = 99 nM T46937 CS6V2F 118711187 IC50 = 142 nM T46937 C4G0NR 118711190 IC50 = 11 nM T46937 C0R4SX 118711191 IC50 = 11 nM T46937 CP9U2T 118711192 IC50 = 336 nM T46937 CU0PB7 118711193 IC50 = 143 nM T46937 C7RFM3 118711194 IC50 = 574 nM T46937 CE37HG 118711247 IC50 = 480 nM T46937 CEWV27 118711248 IC50 = 75 nM T46937 C9UJH0 118711249 IC50 = 266 nM T46937 CCN04Q 118711250 IC50 = 559 nM T46937 CB1L4V 118711969 IC50 = 80 nM T46937 CD3W2I 118711970 IC50 = 17 nM T46937 CD7G9H 118711971 IC50 = 47 nM T46937 C2C6BT 118711972 IC50 = 24 nM T46937 CP32DO 118711973 IC50 = 4000 nM T46937 CU6ZG2 118711974 IC50 = 304 nM T46937 CKR2L7 127038948 IC50 = 730 nM T46937 CBXP14 127038950 IC50 = 1120 nM T46937 CN7C8A 127039315 IC50 = 220 nM T46937 C2N9XI 127039918 IC50 = 210 nM T46937 CF0M8H 127039999 IC50 = 2400 nM T46937 CV8XS2 127040346 IC50 = 140 nM T46937 CIMH26 127040665 IC50 = 1020 nM T46937 C7RQT4 127040675 IC50 = 3100 nM T46937 CNPL48 127040996 IC50 = 9300 nM T46937 CH42ZI 127040998 IC50 = 340 nM T46937 CV4AL5 127041004 IC50 = 1350 nM T46937 C9ON2A 127041006 IC50 > 200000 nM T46937 CKB30T 127041008 IC50 = 156000 nM T46937 CL7VJ2 127047545 IC50 = 8.3 nM T46937 CHIG78 132574706 IC50 = 2340 nM T46937 CMG81E 135434015 EC50 = 100 nM T46937 CE24WD 135838395 EC50 = 6910 nM T46937 C8PHX6 137631406 IC50 = 940000 nM T46937 C6ZB1D 137632198 IC50 = 60.4 nM T46937 CRO8T3 137634506 IC50 = 1260000 nM T46937 CPOU41 137635690 IC50 = 1320000 nM T46937 C7VYP0 137639442 IC50 = 1020000 nM T46937 C4GA0J 137641946 IC50 = 3590 nM T46937 CT92FG 137642967 IC50 = 940000 nM T46937 C7O3US 137643396 IC50 = 2410 nM T46937 C6G7QI 137644622 IC50 = 860000 nM T46937 CUR8V1 137648798 IC50 = 2960 nM T46937 CE5ON3 137649986 IC50 = 1620000 nM T46937 CAC0Y8 137650737 IC50 = 650000 nM T46937 CM8UT3 137651269 IC50 = 1070000 nM T46937 C3A9YO 137651373 IC50 = 930000 nM T46937 C6G8JF 137651603 IC50 = 950000 nM T46937 CK74CY 137652006 IC50 = 910000 nM T46937 CJ69KN 137652138 IC50 = 920000 nM T46937 CJ07WQ 137654461 IC50 = 1040000 nM T46937 CUAT36 137656414 IC50 = 1500000 nM T46937 CVQ2D4 145967492 IC50 = 86 nM T46937 CMCP51 145967502 IC50 = 1100 nM T46937 CTAL93 145967657 IC50 = 190 nM T46937 CYDT13 145967823 IC50 = 1700 nM T46937 CM6QO7 145967859 IC50 = 4500 nM T46937 CE89CL 145968144 IC50 = 14000 nM T46937 CM6D7Y 145968628 IC50 = 1100 nM T46937 CG7N0Z 145969318 IC50 = 22000 nM T46937 CIT74R 145969360 IC50 = 1500 nM T46937 CJ4YR6 145969559 IC50 = 7900 nM T46937 C5GVL6 145969883 IC50 = 2100 nM T46937 C8SMZ3 145970029 IC50 = 4300 nM T46937 CC0QB7 145970199 IC50 = 8600 nM T46937 CN3L2D 145970219 IC50 = 1500 nM T46937 CY5Z4X 145970444 IC50 = 200 nM T46937 CCU54P 145970653 IC50 = 18000 nM T46937 C03KDV 145970872 IC50 = 1900 nM T46937 CLPQ37 145970953 IC50 = 2500 nM T46937 C4XRG5 145971125 IC50 = 270 nM T46937 C7GI9R 145971167 IC50 = 1100 nM T46937 C54YEP 145986354 IC50 = 21000 nM T46937 CG7JW1 145986356 IC50 = 860 nM T46937 CZ3B4C 145987950 IC50 = 150 nM T46937 C6BOT2 145987961 IC50 = 26000 nM T46937 CNP81R 54719874 IC50 = 800 nM T46937 D00BSX 122635 Ki > 10000 nM T46937 D01APA 66855377 Ki = 7.7 nM T46937 D01IEX 44583582 Ki = 24.9 nM T46937 D02TXW 16681707 IC50 = 29 nM T46937 D07MTB 11510579 Ki > 70000 nM T46937 D08DXA 23675622 IC50 = 3120 nM T46937 D09BUG 10207 Ki > 10000 nM T46937 D0B0ZQ 9875920 Ki = 680 nM T46937 D0C0KJ 5280879 EC50 = 1.3 nM T46937 D0KF2P 44126037 Ki = 139 nM T46937 D0N3FL 44157521 Ki = 21 nM T46937 D0P6KN 44457307 IC50 = 34730 nM T77546 D05EAM 4735 Ki = 290 nM T77546 D0V0NL 2146 Ki = 140 nM T77546 CLRO58 127456 Ki = 1700 nM T77546 CQ85DB 6438855 Ki = 200 nM T77546 C9C6LU 10334080 IC50 > 1000000 nM T77546 CCUJ60 10445232 IC50 > 1000000 nM T77546 CY41LT 10445774 IC50 > 1000000 nM T77546 C9X2AQ 10583188 IC50 = 120 nM T77546 CBP6U9 10589155 IC50 > 1000000 nM T77546 CDY0H7 10728071 IC50 = 1000000 nM T77546 C9ILF3 11147919 IC50 = 16000 nM T77546 CUL1G2 11171749 IC50 = 16000 nM T77546 CI2ZB6 11182637 IC50 = 160 nM T77546 CV0MO3 11184629 IC50 = 19000 nM T77546 C7QW3P 11229730 IC50 = 18000 nM T77546 C25MKL 11263687 IC50 = 5000 nM T77546 C9OU4R 11321047 IC50 = 500 nM T77546 CQV28Z 11333471 IC50 = 50000 nM T77546 C3AYC4 11366979 IC50 = 300 nM T77546 COU09A 12655267 IC50 > 100000 nM T77546 CY7MI9 14049939 Ki = 2700 nM T77546 C8O4SL 14983630 Ki = 170 nM T77546 CH56AF 20668674 IC50 > 100000 nM T77546 C92KMP 44345335 Ki = 7100 nM T77546 CMBT65 44387943 IC50 > 100000 nM T77546 CO6A3U 44387955 IC50 > 1000000 nM T77546 C3ZRO0 44387981 IC50 = 61 nM T77546 C2YI1D 44387984 IC50 = 2500 nM T77546 CZJY25 44387994 IC50 = 1000 nM T77546 C2H1UN 44387996 IC50 = 10000 nM T77546 CR1LE3 135432900 Ki = 25000 nM T77546 CA07BI 135465901 Ki = 100000 nM T77546 C8V6MP 135547345 Ki = 5500 nM T77546 C5F1QX 136076500 Ki = 8000 nM T77546 D0B8TJ 2354 Ki = 13 nM T42446 D01AJY 2284 IC50 = 35 nM T42446 D01RBR 130021 IC50 = 38000 nM T42446 D0C9XA 119 IC50 = 25 nM T42446 CGV16B 14113 Ki = 177000 nM T42446 CZS7U8 44600 IC50 = 1770 nM T42446 CZY5M2 685622 Ki = 92000 nM T42446 CH8RL0 4332683 EC50 = 1900 nM T42446 C14BFY 5024764 EC50 = 5370 nM T42446 CW9MS8 6604928 EC50 = 741.31 nM T42446 C9GF0X 10130862 IC50 = 200 nM T42446 C7UK5Q 10132408 IC50 = 18 nM T42446 CLH26M 10419163 IC50 = 280 nM T42446 C9WNM3 14362811 IC50 = 920 nM T42446 C87UMH 14362819 IC50 = 780 nM T42446 CD7V6F 14362824 IC50 = 500 nM T42446 C2Z4GX 14362838 IC50 = 880 nM T42446 CAOK62 14362839 IC50 = 39 nM T42446 CW2UL1 14362840 IC50 = 360 nM T42446 C5VUL6 15603270 EC50 = 870.96 nM T42446 CR2ZU8 19889410 IC50 = 21300 nM T42446 C4ZA6P 23757305 IC50 = 4410 nM T42446 CM01WR 44433820 EC50 = 5011.87 nM T42446 C7UL4T 44433825 EC50 = 4570.88 nM T42446 CSV94A 44433826 EC50 = 2754.23 nM T42446 CZE52B 44433827 EC50 = 3467.37 nM T42446 C96QPG 44433828 EC50 = 1659.59 nM T42446 CFY27E 44433830 EC50 = 1659.59 nM T42446 C5XLV4 44433839 EC50 = 1202.26 nM T42446 CUXT14 44433840 EC50 = 2041.74 nM T42446 CH8UR6 44433842 EC50 = 1659.59 nM T42446 CJMS06 53261132 EC50 = 99300 nM T42446 CGRZ23 71532869 EC50 = 61800 nM T42446 CNC39I 71601649 EC50 > 100000 nM T42446 CN28FE 71601650 EC50 > 100000 nM T42446 CXN32Z 71716205 EC50 = 66900 nM T42446 C6QT8A 71716206 EC50 > 100000 nM T42446 C2HRA1 71717438 EC50 > 100000 nM T42446 C3FZ2O 71718024 EC50 = 40000 nM T42446 CE2H4L 71718648 EC50 = 53500 nM T42446 CHS3M1 71718649 EC50 > 100000 nM T42446 C02RHD 71719256 EC50 = 15900 nM T42446 C4B1MD 71720465 EC50 > 100000 nM T42446 C30YRP 71720467 EC50 > 100000 nM T42446 CN5I0R 122184355 EC50 = 8.6 nM T42446 D02ALQ 86279004 IC50 = 37900 nM T42446 D03KZK 5097016 IC50 = 29 nM T42446 D07BIF 6335948 IC50 = 2.4 nM T42446 D08LFC 5230 IC50 = 6.6 nM T42446 D0AK9X 125917 IC50 = 610 nM T42446 D0H5JW 44602 IC50 = 15 nM T42446 D0N4WZ 9898878 IC50 = 1350 nM T42446 D0S5YH 122150 IC50 = 33000 nM T42446 D0U4HM 5521 EC50 = 500000 nM T42446 D0V0LA 10219532 IC50 = 166 nM T86918 C9QEP1 448828 Ki = 1800000 nM T86918 C6UQJ0 448829 Ki = 25000 nM T86918 C34ELK 449164 Ki = 75 nM T86918 CV0WS2 449165 Ki = 12 nM T86918 CM6CA2 23644309 Ki = 12 nM T86918 C4ES6H 44333048 EC50 = 20 nM T86918 CG9SW2 44333049 EC50 = 3 nM T86918 CDU94X 44333078 IC50 = 0.3 nM T86918 C3XJ9W 73345199 IC50 = 8 nM T86918 CCUJ79 73346731 EC50 = 6 nM T86918 CM76NZ 73346732 EC50 = 22 nM T86918 CQ1ME6 73349806 EC50 = 4 nM T86918 CBC73K 73349808 IC50 = 1 nM T86918 C3QUR8 73351326 EC50 = 50 nM T86918 CFG96R 73351327 EC50 = 20 nM T86918 CU0ZM1 73354298 IC50 = 0.5 nM T86918 C9CW1L 78349960 Ki = 1250 nM T86918 C69QTW 122189583 Ki = 14.3 nM T86918 CTK0D4 122189584 Ki = 41.6 nM T86918 C89YLA 122191023 IC50 = 2590 nM T86918 C2LOE8 122191024 Ki = 14.7 nM T86918 CM06HN 122191026 Ki = 8 nM T86918 C9L2FX 122191027 Ki = 3600 nM T86918 C67END 122191028 Ki = 6100 nM T86918 D01FHK 3086453 EC50 = 0.05 nM T86918 D0R2BA 445248 Ki = 18000000 nM T85309 CT08EI 484751 IC50 = 5900 nM T85309 CA6W3C 1396823 IC50 = 170000 nM T85309 C6HNE1 2246840 IC50 = 187000 nM T85309 C8O4KD 5281599 IC50 = 17100 nM T85309 C3ZJ8U 5281609 IC50 = 11500 nM T85309 CQEL68 6055630 IC50 = 108000 nM T85309 C9HJE6 7032560 IC50 = 125000 nM T85309 CSJ73Q 10347674 IC50 = 5500 nM T85309 CP2D3Q 10364369 IC50 = 7400 nM T85309 C3MZ0D 14186891 IC50 = 8100 nM T85309 CJ26AL 21604873 IC50 = 83000 nM T85309 CS56LP 49822436 IC50 = 6200 nM T85309 CO87MN 118729943 IC50 = 87000 nM T85309 C09ING 118729944 IC50 = 136000 nM T85309 CD0L9T 145958807 IC50 = 7800 nM T85309 D01BTV 286 IC50 = 1000 nM T85309 D0I4NN 14056555 IC50 = 156000 nM T85309 D0T3PW 5281672 IC50 = 18800 nM T86385 D00UVA 11556711 IC50 > 30000 nM T86385 D0FT4R 107706 IC50 > 10000 nM T86385 D0SH3I 387447 IC50 = 520 nM T86385 D00LOB 9866964 Ki > 26000 nM T86385 D01YIO 10146470 Ki = 38 nM T86385 D0VO0T 24800541 EC50 = 13.5 nM T86385 D0Y6SQ 2536 IC50 > 100000 nM T86385 D0HM5J 118253852 IC50 > 20000 nM T86385 D0NJ1A 65663 IC50 = 1100 nM T86385 D0WY9H 9892148 Ki = 250 nM T86385 CKO7V4 1701 IC50 = 250000 nM T86385 CP9FG4 99625 IC50 = 24000 nM T86385 CLX4V7 130395 IC50 > 100000 nM T86385 C5Q7EX 160817 IC50 > 60000 nM T86385 CC9E0Y 232547 IC50 = 2100 nM T86385 CN0XJ3 439647 IC50 = 110000 nM T86385 CN67CR 555078 IC50 = 3700 nM T86385 CHF5A4 578663 IC50 = 433200 nM T86385 C05EGK 736344 IC50 > 1000000 nM T86385 CW9DQ2 4476325 IC50 = 4100 nM T86385 CHU41D 5013064 IC50 > 60000 nM T86385 CF9VK2 5236960 IC50 > 139000 nM T86385 CO58XD 5311161 IC50 > 100000 nM T86385 C8OE6S 6913584 IC50 > 100000 nM T86385 CANW64 9798519 IC50 = 700 nM T86385 CMUY79 9800909 IC50 = 52 nM T86385 CD8G1T 9818360 IC50 = 4500 nM T86385 C9NHA3 9821476 IC50 = 1500 nM T86385 C7UKF5 9825353 IC50 > 1000 nM T86385 C3K8PQ 9830518 IC50 = 530 nM T86385 CGNB60 9830581 IC50 = 280 nM T86385 CL61HY 9888442 IC50 > 100000 nM T86385 CG2EZ0 9889108 IC50 < 100000 nM T86385 C5T0GJ 9895523 IC50 = 64 nM T86385 C7KJP3 9908917 IC50 > 100000 nM T86385 CGL12S 9916581 Ki = 1390 nM T86385 CQ84MG 9917430 Ki > 600000 nM T86385 CGT3K4 9932145 IC50 > 100000 nM T86385 CIQX83 9938207 Ki = 379 nM T86385 C2CE1A 9962331 Ki > 2000000 nM T86385 C3HI6E 9972080 IC50 > 100000 nM T86385 C0WT4P 10024711 IC50 = 20000 nM T86385 CVHQ60 10048700 Ki = 130000 nM T86385 C7CW1P 10080504 IC50 = 740 nM T86385 CEN06H 10093642 IC50 > 100000 nM T86385 CD6KX7 10162462 IC50 > 1000 nM T86385 CRP54X 10364794 IC50 = 22000 nM T86385 C9M3VF 10366027 IC50 > 1000 nM T86385 CCQA34 10383086 IC50 > 1000000 nM T86385 C79FQG 10383359 Ki = 400000 nM T86385 CEPM12 10391460 IC50 = 8.4 nM T86385 CCL85B 10394816 IC50 = 1.4 nM T86385 C2UNX1 10407325 IC50 = 3700 nM T86385 CORP79 10431323 IC50 > 100000 nM T86385 C9M7CE 10497407 IC50 = 330 nM T86385 CYC5G6 10497621 IC50 = 220 nM T86385 CJN97A 10499538 IC50 = 1700 nM T86385 C6D3UM 10504812 IC50 = 83000 nM T86385 CA4RW1 10517868 IC50 > 60000 nM T86385 COKF15 10520443 IC50 = 4500 nM T86385 CIMX79 10524714 IC50 = 600 nM T86385 C5LR1J 10527210 IC50 = 4800 nM T86385 C3VQM6 10529952 IC50 = 200 nM T86385 CTN78E 10545533 IC50 = 4200 nM T86385 CCE5M4 10551184 IC50 = 4800 nM T86385 CZL85V 10572734 IC50 > 100000 nM T86385 CVO85L 10577862 IC50 = 440000 nM T86385 C20JKT 10593313 IC50 = 780 nM T86385 CZ8PK9 10599803 IC50 = 2300 nM T86385 C2V4IZ 10616405 IC50 = 100000 nM T86385 C9I3QE 10616695 IC50 = 1500 nM T86385 CS52KZ 10617888 IC50 = 2200 nM T86385 C38SDV 10619385 IC50 = 340 nM T86385 C83JQD 10620089 IC50 = 230 nM T86385 C4K1BD 10620298 IC50 = 6500 nM T86385 C5X0QT 10625780 IC50 = 77 nM T86385 C6V4NJ 10642042 IC50 = 75000 nM T86385 CBHW74 10653967 Ki > 15000 nM T86385 CMXS14 10653995 Ki > 15000 nM T86385 CM57UY 10666214 IC50 = 1900 nM T86385 C8QB4K 10689926 IC50 = 6500 nM T86385 CZ57RO 10697572 IC50 = 6600 nM T86385 C6S2JY 10712874 IC50 = 2500 nM T86385 CFCP28 10714430 IC50 = 640 nM T86385 CP7Y9Z 10714544 IC50 = 4100 nM T86385 CPT0M6 10715096 IC50 = 3900 nM T86385 CE7CB3 10715299 IC50 = 5400 nM T86385 CD0I2U 10736348 IC50 = 8000 nM T86385 CX9JY3 10737216 IC50 = 1000 nM T86385 C06EQF 10739429 IC50 > 100000 nM T86385 CVX58I 10740202 IC50 = 3700 nM T86385 C1TB8N 10764081 IC50 > 100000 nM T86385 C3MH6G 10765640 IC50 = 16000 nM T86385 C4J2AM 10782637 IC50 = 1800 nM T86385 CSO9H0 10811389 IC50 > 100000 nM T86385 CG9B1J 10819798 Ki > 15000 nM T86385 CL85VD 10835279 IC50 = 3300 nM T86385 CX3E7A 10838826 IC50 = 1500 nM T86385 C39NQW 11235804 Ki = 9500 nM T86385 C92PMV 11253808 IC50 = 55000 nM T86385 CLAK97 11540629 IC50 = 16000 nM T86385 C93USP 11626693 IC50 = 2900 nM T86385 C07MTY 11634767 IC50 = 28000 nM T86385 C1ZK9V 11684537 IC50 = 8000 nM T86385 C6RY7J 11725023 IC50 = 80000 nM T86385 CC53TD 12043588 IC50 = 63000 nM T86385 C10ALY 13339657 IC50 = 32000 nM T86385 C2DGN3 14046022 IC50 = 3100 nM T86385 CDP91C 15743471 IC50 > 60000 nM T86385 CJ41CN 15743472 IC50 = 25000 nM T86385 C9OSM6 16144480 Ki > 15000 nM T86385 CDR0G7 16145606 Ki > 15000 nM T86385 CY20PW 16147332 Ki > 15000 nM T86385 CF5Y3L 16147570 Ki > 15000 nM T86385 C7S6IT 16148231 Ki = 1500 nM T86385 C63HAE 18572952 IC50 > 134000 nM T86385 CZPF48 23648277 IC50 > 50000 nM T86385 C1Z9SX 24776379 Ki = 0.15 nM T86385 CN0VA7 24822701 IC50 > 50000 nM T86385 CCG0Z2 25124204 IC50 = 22 nM T86385 CUC8N5 25141405 IC50 > 100000 nM T86385 C3GS6F 33009902 IC50 > 10000 nM T86385 CL0M7R 44143089 IC50 = 147910.84 nM T86385 C8Y9JZ 44284991 Ki = 44.1 nM T86385 CMZ71H 44284992 Ki = 3.74 nM T86385 C5NU9L 44285118 Ki = 14.3 nM T86385 CU9G2F 44285211 Ki = 0.916 nM T86385 C0FPN1 44285253 Ki = 25.3 nM T86385 C9N1ZL 44285281 Ki = 0.187 nM T86385 C5PX3O 44285312 Ki = 0.174 nM T86385 C9LRW8 44285352 Ki = 3.85 nM T86385 CN7SA3 44287645 IC50 = 33000 nM T86385 C1GU7P 44287670 IC50 = 56000 nM T86385 CB8L9Q 44287782 IC50 = 37000 nM T86385 CR6QO0 44287881 IC50 > 60000 nM T86385 CT98XO 44287910 IC50 = 55000 nM T86385 C4KWZ8 44287967 IC50 = 24000 nM T86385 C6KJ4D 44288060 IC50 > 60000 nM T86385 CMO3X2 44288136 IC50 = 28000 nM T86385 C65TOU 44303193 IC50 = 17000 nM T86385 C2DM3E 44303204 IC50 = 12000 nM T86385 C9N4KA 44303215 IC50 = 11000 nM T86385 CE3NJ0 44303216 IC50 = 210000 nM T86385 C3E6HC 44303217 IC50 = 9300 nM T86385 CR68VO 44303218 IC50 = 65000 nM T86385 CR6GO9 44303240 IC50 = 91000 nM T86385 C6YB7J 44303242 IC50 = 25000 nM T86385 CWOM61 44303259 IC50 = 8100 nM T86385 C0C8FX 44303260 IC50 = 23000 nM T86385 CWUI78 44303375 IC50 = 18000 nM T86385 CJ15HX 44303391 IC50 = 58000 nM T86385 CH6TE7 44303392 IC50 = 24000 nM T86385 CVJS18 44303415 IC50 = 25000 nM T86385 C1W6MX 44303477 IC50 = 42000 nM T86385 CSB6M5 44303496 IC50 = 12000 nM T86385 CGNR45 44303533 IC50 = 890000 nM T86385 CTRX10 44303534 IC50 = 130000 nM T86385 C20OYT 44303535 IC50 = 36000 nM T86385 C1Y2QB 44303536 IC50 = 140000 nM T86385 CGP52Y 44303588 IC50 = 35000 nM T86385 CH13CK 44303589 IC50 = 32000 nM T86385 CQ82JC 44303644 IC50 = 30000 nM T86385 CO3V6E 44303657 IC50 = 44000 nM T86385 C5L1DC 44308976 IC50 > 100000 nM T86385 CKN8C1 44316486 IC50 = 230 nM T86385 C2AT7J 44342409 Ki > 15000 nM T86385 CD8AL2 44351097 IC50 = 3600 nM T86385 CHGE39 44351104 IC50 = 67000 nM T86385 CQH2K6 44353359 Ki = 200 nM T86385 C14NKU 44353376 Ki = 1600 nM T86385 CK13HZ 44353387 Ki = 1100 nM T86385 C4OQZ5 44353439 Ki = 200 nM T86385 CDLQ89 44354931 IC50 = 75 nM T86385 CZG9E2 44354934 IC50 = 170 nM T86385 C7NWU8 44354935 IC50 = 1600 nM T86385 C5UJB8 44354936 IC50 = 6.4 nM T86385 CRL78E 44354968 IC50 = 520 nM T86385 CM73HF 44354971 IC50 = 160 nM T86385 CVYF38 44354984 IC50 = 140 nM T86385 CZDW93 44355000 IC50 = 15 nM T86385 CG1VN6 44355001 IC50 = 190 nM T86385 CL04TR 44355071 IC50 = 69 nM T86385 C9U4BR 44355072 IC50 = 48 nM T86385 CI4R1U 44355083 IC50 = 80 nM T86385 CDON50 44355100 IC50 = 21000 nM T86385 C34UGZ 44366594 Ki = 1700 nM T86385 CFL1J0 44366665 Ki > 1000000 nM T86385 C27VSQ 44366666 Ki = 2200 nM T86385 CNE14G 44378491 IC50 = 500 nM T86385 CSV48N 44378519 IC50 = 380 nM T86385 CL9HZ0 44378543 IC50 = 800 nM T86385 CDA68B 44378603 IC50 = 1300 nM T86385 C34YAJ 44378694 IC50 = 1000 nM T86385 C3BX5Y 44412781 Ki > 150000 nM T86385 CIT5G7 44561891 IC50 > 100000 nM T86385 C90BGR 44561892 IC50 > 100000 nM T86385 C9RGX4 44561893 IC50 > 100000 nM T86385 CU7NP5 44561930 IC50 > 100000 nM T86385 CV21IQ 44561931 IC50 > 100000 nM T86385 CR08WA 44561932 IC50 > 100000 nM T86385 C2PVE0 45103523 Ki > 26000 nM T86385 CGN14R 45103723 Ki > 26000 nM T86385 CD4T1L 46221636 IC50 = 120000 nM T86385 CUI91D 46905615 IC50 = 1200 nM T86385 CJH50R 49797481 IC50 > 100000 nM T86385 CI7P2B 49797571 IC50 = 90 nM T86385 CI59MV 49797572 IC50 > 50000 nM T86385 C96CKU 49797573 IC50 = 150 nM T86385 CEC3R4 52943167 IC50 = 100 nM T86385 C5H3GD 52943168 IC50 = 200 nM T86385 C4WVX9 52943169 IC50 = 200 nM T86385 C8AR2B 52946468 IC50 = 100 nM T86385 CZ3FS0 52949270 IC50 = 150 nM T86385 CO6F3U 53249965 IC50 = 1400 nM T86385 CBJQ98 54132077 IC50 = 53000 nM T86385 CY3IO1 56659828 IC50 > 10 nM T86385 CI2AB4 56663296 IC50 > 10 nM T86385 CT2G3R 56666720 IC50 = 2.1 nM T86385 CQH46K 56666721 IC50 > 10 nM T86385 C3V0AU 56666722 IC50 > 10 nM T86385 CZ3O2H 56670144 IC50 > 10 nM T86385 CNL70Y 56670149 IC50 = 7 nM T86385 C0HJL7 56673658 IC50 = 4.8 nM T86385 CP5B7A 56673659 IC50 = 8.8 nM T86385 CE58OY 56673664 IC50 > 10 nM T86385 C9F5UR 56676983 IC50 > 10 nM T86385 CL9XA8 56680306 IC50 > 10 nM T86385 CHNX69 56680307 IC50 > 10 nM T86385 CP3IV1 56680314 IC50 > 10 nM T86385 CSF9P8 56683631 IC50 > 10 nM T86385 CD57KP 56683632 IC50 > 10 nM T86385 CP1MR2 56683633 IC50 > 10 nM T86385 CG7O3N 56683634 IC50 = 9.5 nM T86385 CL16UQ 56949326 IC50 < 10000 nM T86385 C0UIF5 57671050 IC50 = 7800 nM T86385 CY26NE 57671116 IC50 > 10000 nM T86385 C9E6CB 57671131 IC50 > 10000 nM T86385 CJO75X 57671161 IC50 = 8500 nM T86385 CF2Q3E 59497392 IC50 > 10000 nM T86385 C2W3AK 59497404 IC50 > 10000 nM T86385 C0E1KN 59497528 IC50 = 5400 nM T86385 CAWN80 59497611 IC50 > 10000 nM T86385 CSQY41 59497643 IC50 > 10000 nM T86385 C31NTK 59497690 IC50 > 10000 nM T86385 C48UHX 66561877 IC50 = 369000 nM T86385 C50MEH 71682307 IC50 > 10000 nM T86385 CO8PQ5 71682308 IC50 = 3800 nM T86385 C78DJQ 71711730 IC50 < 10000 nM T86385 CL23VT 71723878 IC50 = 16000 nM T86385 C1MBU7 72793747 IC50 > 100000 nM T86385 C6BY5D 72793776 IC50 > 100000 nM T86385 C1DI8A 72793778 IC50 = 19000 nM T86385 C5U9CI 73355715 Ki = 0.437 nM T86385 CFPT98 90655054 IC50 > 30000 nM T86385 C5JZ8R 90655055 IC50 > 30000 nM T86385 C8E4WS 102323332 IC50 > 50000 nM T86385 CR2AU7 118010068 IC50 > 10000 nM T86385 COA36C 118010069 IC50 > 10000 nM T86385 C5NJH1 118202505 IC50 > 10000 nM T86385 C43ADS 118202506 IC50 > 10000 nM T86385 C2UXT7 118202507 IC50 > 10000 nM T86385 CPV27G 118202509 IC50 > 10000 nM T86385 CJB3K7 118202510 IC50 > 10000 nM T86385 C12BHL 118202511 IC50 > 10000 nM T86385 COT6H0 118202512 IC50 > 10000 nM T86385 C0GRU4 118718129 Ki = 3.9 nM T86385 C8ZSC2 118727248 IC50 > 10000 nM T86385 CYIX41 118727249 IC50 > 10000 nM T86385 CH1T3M 118727250 IC50 > 10000 nM T86385 CVG1X5 118727251 IC50 > 10000 nM T86385 C9B6KX 118727252 IC50 > 10000 nM T86385 C3OUW6 118727253 IC50 > 10000 nM T86385 C10QJC 118727254 IC50 > 10000 nM T86385 CVIF56 118727255 IC50 > 10000 nM T86385 CNQ9U4 118727256 IC50 > 10000 nM T86385 CN93WU 118727257 IC50 > 10000 nM T86385 C5DR7Z 118727258 IC50 > 10000 nM T86385 CDEU05 118727259 IC50 > 10000 nM T86385 CZHT12 118727260 IC50 > 10000 nM T86385 CD21PC 118731187 IC50 = 6000 nM T86385 CGV2Y0 122192762 Ki = 12 nM T86385 C6RDX4 122192767 Ki = 490 nM T86385 C9QKI3 127020966 IC50 > 100000 nM T86385 CNL2Z9 137635679 Ki = 0.89 nM T86385 CDQ62V 137637214 Ki > 50000 nM T86385 C2K8JV 137639385 Ki > 50000 nM T86385 CNO8Y2 137639848 Ki = 3.4 nM T86385 CCF5A0 137640149 Ki = 4.8 nM T86385 CZ95CD 137642316 Ki = 62 nM T86385 CF0TK8 137642520 Ki = 7.3 nM T86385 C8WS7U 137646736 Ki = 390 nM T86385 CCQ4H7 137647098 Ki = 1200 nM T86385 C03IMN 137647139 Ki = 1.7 nM T86385 C71MRD 137649122 Ki = 160 nM T86385 C2D6KY 137650380 Ki = 410 nM T86385 CYGV01 137650976 Ki = 1.1 nM T86385 COR29F 137652632 Ki = 480 nM T86385 CNX46H 137654508 Ki > 50000 nM T86385 CZ1H4R 137655362 Ki = 1.6 nM T86385 CQAV71 137657536 Ki = 12 nM T86385 CD25CQ 137657864 Ki = 530 nM T86385 CTUM82 137658421 IC50 = 1100 nM T86385 CIGV31 137660044 Ki = 630 nM T86385 C1S2LC 137660418 Ki = 3000 nM T86385 CX5S3Y 137661570 Ki = 4.9 nM T86385 CE7GI1 137662261 Ki = 2.9 nM T86385 CYT20V 155514020 Ki = 29000 nM T86385 CW1B5Z 155521967 Ki < 0.1 nM T86385 CBU5W0 155524880 IC50 > 10000 nM T86385 C4QT3M 155526246 Ki = 54 nM T86385 C2X5EJ 155531124 Ki = 160 nM T86385 CPC60R 155533917 Ki = 7.4 nM T86385 CM06WG 155535720 Ki = 38 nM T86385 CU9FL4 155551858 Ki = 13000 nM T86385 C2E5GR 155554478 IC50 > 10000 nM T86385 CE3G5W 155556110 Ki = 1200 nM T86385 C0SND3 155557259 Ki = 5200 nM T86385 CTS63Q 155558248 Ki = 150 nM T86385 CFX07G 155558369 IC50 > 5000 nM T86385 C5R4VY 155566937 Ki = 8.2 nM T86385 CP4F1U 155567613 Ki = 7800 nM T86385 CU42CE 155567829 IC50 > 100000 nM T86385 CO8GJ3 155568502 Ki = 14 nM T86385 CU62EW 155568945 Ki = 0.26 nM T86385 D02AVL 18376720 Ki > 5000 nM T86385 D02PAU 16731825 Ki > 10000 nM T86385 D05ICF 3492365 IC50 = 2.3 nM T86385 D08QZD 9829503 Ki = 720 nM T86385 D0C1NP 66561876 IC50 = 14200 nM T86385 D0E9EH 44353386 Ki > 800000 nM T86385 D0F2YC 10038543 IC50 = 0.39 nM T86385 D0F3CA 1609 IC50 = 93000 nM T86385 D0R9CH 3400921 Ki > 10000 nM T09185 D00STL 644241 IC50 < 100 nM T09185 D0AZ3C 5291 IC50 = 43 nM T09185 D0E6XR 3062316 IC50 = 0.5 nM T09185 D0E3TC 44259 IC50 = 4.28 nM T09185 D0D5PL 71577234 IC50 = 164 nM T09185 D0LL1P 71768628 IC50 = 97 nM T09185 CL14BG 4426513 IC50 > 100000 nM T09185 CA3I4T 24753787 IC50 > 50000 nM T09185 CJ0CU5 24825841 IC50 = 2.4 nM T09185 C4FZ8E 24875320 IC50 = 4.799 nM T09185 C3VRO9 44557921 IC50 > 10000 nM T09185 CF57GK 46215462 IC50 = 20 nM T09185 C2VAX9 51035420 IC50 = 68 nM T09185 CPHX64 57325478 IC50 > 50000 nM T09185 CQ9BW4 57325479 IC50 > 50000 nM T09185 CVK0G4 58056356 IC50 > 50000 nM T09185 C7SGT6 60202316 IC50 = 39 nM T09185 CV63UL 67240318 IC50 > 10000 nM T09185 CB61ZO 67347910 IC50 = 9 nM T09185 CRH2Y9 68639605 IC50 = 8.93 nM T09185 C1IT5U 71550931 IC50 = 6.8 nM T09185 CG1I5B 71550932 IC50 = 7.02 nM T09185 C1F5NV 71624671 IC50 = 39.63 nM T09185 CQE01I 71624672 IC50 = 65.14 nM T09185 CV8XI0 71624673 IC50 > 1000 nM T09185 CY82NR 71624674 IC50 = 29.15 nM T09185 C0IM7Z 71624675 IC50 = 39.82 nM T09185 C6JS8P 71624676 IC50 = 38.9 nM T09185 C2F0QN 71624677 IC50 > 1000 nM T09185 CQ75IY 71624788 IC50 = 5.96 nM T09185 C6GT1Q 71624789 IC50 = 47.75 nM T09185 C6ZYR9 71624790 IC50 > 1000 nM T09185 CCSI30 71624792 IC50 > 1000 nM T09185 C4JD7I 71624793 IC50 = 470 nM T09185 CS0AQ6 71624904 IC50 = 4.04 nM T09185 C23XIU 71624905 IC50 = 22.36 nM T09185 C4KTH9 71624906 IC50 = 16.64 nM T09185 C7BG9F 71624907 IC50 = 19.75 nM T09185 CC61DF 71624908 IC50 = 6.14 nM T09185 CRLN56 71624909 IC50 > 1000 nM T09185 CLO8V2 71625035 IC50 = 35.02 nM T09185 CQI0N1 71625036 IC50 = 9.72 nM T09185 CO41GB 71625037 IC50 = 19.03 nM T09185 CC68IJ 71625038 IC50 = 386.5 nM T09185 C4SV3X 71625039 IC50 = 324.1 nM T09185 CT2K6M 71625040 IC50 = 6.34 nM T09185 C6JZ2E 71625161 IC50 = 29.81 nM T09185 CRGQ64 71625290 IC50 = 6.71 nM T09185 CP83JY 71625291 IC50 = 13.94 nM T09185 CGJ8H4 71625292 IC50 = 13.3 nM T09185 C0D4LN 71625406 IC50 = 17.49 nM T09185 C9B1RV 71625407 IC50 = 37.58 nM T09185 CKOL80 71625408 IC50 = 12.47 nM T09185 CQY4U2 71625409 IC50 = 10.05 nM T09185 C42VJY 71764060 IC50 = 235 nM T09185 CEH2B7 72836888 IC50 = 86 nM T09185 C9IZF3 86763814 IC50 = 1500 nM T09185 CR9V4A 86763924 IC50 = 6 nM T09185 C6F5PQ 119081684 IC50 = 309 nM T09185 CN4X0C 121231414 IC50 = 9.4 nM T09185 C81IFQ 122163152 IC50 = 2110 nM T09185 C49UGP 122187122 IC50 = 150 nM T09185 CQL0W7 122197565 IC50 = 75.7 nM T09185 C6UY2L 122633880 IC50 = 212 nM T09185 CC7P2W 122633900 IC50 = 265 nM T09185 CN41IF 122634050 IC50 = 292 nM T09185 CBYC49 126617676 IC50 = 22.2 nM T09185 CC58IQ 127043948 IC50 = 126 nM T09185 CVF8Z9 127045862 IC50 = 4.7 nM T09185 CH68NT 127046076 IC50 = 137 nM T09185 CF5D2Y 129318936 IC50 = 2462 nM T09185 C6RPF1 130364436 IC50 = 191 nM T09185 CSY34O 130364443 IC50 = 254 nM T09185 CI9H2W 130364450 IC50 = 24.3 nM T09185 CM4TO5 130364451 IC50 = 38.3 nM T09185 C28CLN 130364457 IC50 = 328 nM T09185 CV4DH7 130364460 IC50 = 80.7 nM T09185 CW91ZV 130364461 IC50 = 223 nM T09185 CQIZ43 130364463 IC50 = 89 nM T09185 C4IKC6 130364464 IC50 = 123 nM T09185 C0X6JS 130364465 IC50 = 79.9 nM T09185 C0ZGC1 130364467 IC50 = 71.1 nM T09185 CO9C5Q 130364468 IC50 = 442 nM T09185 CQW3P1 130364471 IC50 = 50.5 nM T09185 CHWX05 130364473 IC50 = 49.9 nM T09185 CLB65Y 130364478 IC50 = 66.6 nM T09185 CUZG19 130364481 IC50 = 614 nM T09185 C34OMJ 130364482 IC50 = 209 nM T09185 C6TWR3 130364484 IC50 = 132 nM T09185 C8SF5Q 130364488 IC50 = 19.9 nM T09185 CS5C4E 130364494 IC50 = 222 nM T09185 CVQ32Y 130364503 IC50 = 25.6 nM T09185 CV8B0Y 130364506 IC50 = 545 nM T09185 CHX23J 130364524 IC50 = 44.6 nM T09185 CHYL89 130364535 IC50 = 167 nM T09185 C6OMB1 132204257 IC50 = 63 nM T09185 C6ROQ3 132546210 IC50 = 116 nM T09185 CQR94G 134198433 IC50 = 193 nM T09185 C1X6FJ 134693894 IC50 = 9.4 nM T09185 CXC69T 137321158 IC50 = 35 nM T09185 CWC49K 137321210 IC50 = 5.6 nM T09185 CI1E8V 137634241 IC50 > 10000 nM T09185 C5VE4K 137636547 IC50 = 167 nM T09185 CZ05TY 137637593 IC50 = 10000 nM T09185 CU9YQ3 137637635 IC50 = 5020 nM T09185 C6PKY7 137645383 IC50 > 10000 nM T09185 CHR9E0 137651685 IC50 = 13.1 nM T09185 CY53VO 137651787 IC50 > 10000 nM T09185 CE8DW7 137658399 IC50 > 10000 nM T09185 CU61WM 137658936 IC50 > 10000 nM T09185 CY9N8Q 137662234 IC50 = 6.6 nM T09185 C3K5LU 137796291 IC50 = 326 nM T09185 CM3A8O 139030333 IC50 = 3000 nM T09185 C6AK0N 139030518 IC50 = 135 nM T09185 CB69CL 145925694 IC50 = 0.7078 nM T09185 C7SH9V 145949579 IC50 = 3.2 nM T09185 CQCV54 145950906 IC50 = 151 nM T09185 CKWZ34 145950923 IC50 = 6.2 nM T09185 CGOE73 145951398 IC50 = 11.4 nM T09185 CZF70O 145951916 IC50 = 5 nM T09185 CNK12Z 145952731 IC50 = 12.5 nM T09185 CGV16H 145954003 IC50 = 1200 nM T09185 CUIT87 145955254 IC50 = 7.9 nM T09185 CX2U6N 145956375 IC50 = 16 nM T09185 CC0RU9 145956925 IC50 = 614 nM T09185 CA2F0O 145958559 IC50 = 3.9 nM T09185 C12VOP 145959821 IC50 = 380 nM T09185 C5PZ9J 145959874 IC50 = 8.4 nM T09185 CF0C6K 145960274 IC50 = 3.9 nM T09185 CQE9M5 145966810 IC50 = 100 nM T09185 CWJ12M 145969155 IC50 = 35 nM T09185 C8NDS6 145971939 IC50 = 12.6 nM T09185 CP9NB6 145974090 IC50 = 695 nM T09185 CI85EU 145998085 IC50 = 14.9 nM T09185 CD49VM 155295006 IC50 = 23.8 nM T09185 CSHC63 155510467 IC50 = 359.5 nM T09185 C5MP1Q 155510890 IC50 = 36.4 nM T09185 CG09WO 155512858 IC50 = 55.6 nM T09185 C6H8ZU 155513172 IC50 = 10.4 nM T09185 CZDH58 155514096 IC50 = 36.5 nM T09185 CDU75B 155514157 IC50 = 3.97 nM T09185 CB5T9G 155515436 IC50 = 15.5 nM T09185 CUHZ87 155516883 IC50 = 723.1 nM T09185 C84GJO 155517474 IC50 = 21.3 nM T09185 C63PZX 155518871 IC50 = 42.3 nM T09185 CT0V6H 155519724 IC50 = 10.5 nM T09185 CNP8T7 155530083 IC50 = 9.2 nM T09185 CK10UA 155531677 IC50 = 16.5 nM T09185 CS69CA 155532132 IC50 = 3 nM T09185 CURO30 155532620 IC50 = 5.89 nM T09185 C3PWI1 155534046 IC50 > 1000 nM T09185 CWLZ25 155535008 IC50 = 107.8 nM T09185 CTXK93 155535665 IC50 = 14.4 nM T09185 C14SEB 155535950 IC50 = 42.5 nM T09185 C8NA6L 155536370 IC50 = 8.7 nM T09185 CPG5T4 155538560 IC50 > 3000 nM T09185 C3O6WX 155540330 IC50 > 1000 nM T09185 CXG71B 155540768 IC50 = 36.4 nM T09185 C3Q9UA 155541932 IC50 = 1260 nM T09185 C76NKG 155543431 IC50 = 68.7 nM T09185 CC9LQ2 155546287 IC50 = 13000 nM T09185 CI27QV 155546853 IC50 = 4879 nM T09185 CYP2O5 155547984 IC50 = 63.7 nM T09185 C9MJL5 155551408 IC50 = 14.7 nM T09185 C14QWH 155551649 IC50 > 3000 nM T09185 CL8KR2 155552517 IC50 = 357.1 nM T09185 CA9Y3J 155552522 IC50 = 8.53 nM T09185 C1TA9J 155553503 IC50 = 73.8 nM T09185 C8BAU3 155554243 IC50 = 92 nM T09185 CCQF25 155555943 IC50 = 22.5 nM T09185 C7N1AT 155560186 IC50 > 2000 nM T09185 CYD1C7 155560599 IC50 > 1000 nM T09185 C2EDK1 155562180 IC50 = 15.2 nM T09185 C2QC5F 155562643 IC50 > 1000 nM T09185 CHLY93 155562871 IC50 = 30.3 nM T09185 CBG9Z1 155562952 IC50 = 150.5 nM T09185 C0WZ9S 155563842 IC50 > 1000 nM T09185 C60KLJ 155564326 IC50 = 1296 nM T09185 C4BS6J 155565938 IC50 = 15.6 nM T09185 CINX89 155566065 IC50 = 4850 nM T09185 C7Q4RY 155566792 IC50 = 30.1 nM T09185 C0V7SM 155567015 IC50 = 638.9 nM T09185 CP69SU 155567937 IC50 = 66.9 nM T09185 D0BL0O 71624791 IC50 = 2.29 nM T30803 D00ENY 33032 Ki = 42700 nM T30803 D01OXI 2578 IC50 = 8100 nM T30803 D03GET 4055 Ki = 12100 nM T30803 D04OSE 4485 Ki = 17400 nM T30803 D0K8KX 5280343 IC50 = 218000 nM T30803 D0V4GY 9552079 Ki = 192000 nM T30803 C52MFS 1756 IC50 > 50000 nM T30803 CBF49Z 7416 Ki = 274100 nM T30803 CT48KR 21025 IC50 = 79300 nM T30803 CRT9K5 128254 IC50 < 1000 nM T30803 CCZ04P 214232 IC50 = 105000 nM T30803 C8MEI0 223143 IC50 = 20300 nM T30803 CB1K8N 363243 IC50 = 5000 nM T30803 CUF5O9 390735 IC50 > 50000 nM T30803 CJKN12 432139 IC50 = 64800 nM T30803 CN1TR3 580286 IC50 > 173000 nM T30803 C39UQA 723918 IC50 > 212000 nM T30803 CTX3F0 831028 IC50 > 157000 nM T30803 C2ZL6W 877340 IC50 = 86300 nM T30803 CV0S1M 877450 IC50 = 58000 nM T30803 C4L7CX 1550330 IC50 > 100000 nM T30803 C39ODA 1550696 IC50 > 100000 nM T30803 CD4IA9 1712537 IC50 > 155000 nM T30803 CK1N3W 2223018 IC50 > 135000 nM T30803 C2O8ZG 2288440 IC50 = 24900 nM T30803 C4VJW9 2724179 Ki = 211 nM T30803 C1ESQ4 2862129 IC50 > 100000 nM T30803 C49TLS 2881754 IC50 > 100000 nM T30803 C07WHI 4362773 IC50 > 100000 nM T30803 CSZU71 4448737 IC50 = 20400 nM T30803 CHW3L7 5291033 IC50 > 100000 nM T30803 C9ZG4E 5325382 IC50 > 50000 nM T30803 C8VZ9T 5325386 IC50 > 50000 nM T30803 C1BM9S 5377539 IC50 > 100000 nM T30803 C0MPR9 5387357 IC50 > 100000 nM T30803 CZT90E 5802828 IC50 > 100000 nM T30803 CW0E3Y 5925463 IC50 > 100000 nM T30803 C4VK5N 6382486 IC50 > 100000 nM T30803 CC92GK 6445552 IC50 > 100000 nM T30803 C3MX1J 9979274 IC50 = 20000 nM T30803 C6XJT3 10026610 IC50 = 40000 nM T30803 CR95VY 10072380 IC50 = 44700 nM T30803 C35RWB 10253825 IC50 = 55800 nM T30803 CKJO89 10317614 IC50 = 3500 nM T30803 CB2D6A 10319412 IC50 = 18000 nM T30803 C4US6F 10387232 IC50 = 14000 nM T30803 CRYV80 10429818 IC50 = 2500 nM T30803 C8T6XZ 10475024 IC50 = 12000 nM T30803 CI2B1P 10489510 IC50 = 12300 nM T30803 CAJ5W4 10791392 Ki = 2000000 nM T30803 CD8WK2 10847727 IC50 = 18900 nM T30803 C9NC5T 10964817 IC50 = 21000 nM T30803 CI2T6R 11595259 IC50 = 4.1 nM T30803 CK2Y6S 11798906 Ki = 2200000 nM T30803 CG1CU7 12219475 IC50 > 50000 nM T30803 C4EUP9 12247627 IC50 = 2000 nM T30803 CLK87P 13989170 IC50 = 2000 nM T30803 C62BRX 14016406 IC50 < 1000 nM T30803 CJ4OE6 14860354 IC50 = 1000 nM T30803 CROS94 15192338 IC50 = 1000 nM T30803 CY32OJ 15192339 IC50 = 3500 nM T30803 CGH65T 15192340 IC50 = 7000 nM T30803 CY3HI1 15192341 IC50 = 8000 nM T30803 CUHY70 15192342 IC50 = 100000 nM T30803 CHX2S0 15192343 IC50 = 25000 nM T30803 CL21QK 15192344 IC50 = 3000 nM T30803 C3F6KS 15192393 IC50 = 8000 nM T30803 C1TS7N 15192395 IC50 = 1000 nM T30803 CD0CS6 15605637 IC50 > 100000 nM T30803 C1V6AR 16047174 IC50 > 100000 nM T30803 C1NQ6R 16047175 IC50 > 100000 nM T30803 C5FS1M 16047278 IC50 > 100000 nM T30803 CYT94W 16047279 IC50 > 100000 nM T30803 CB78XP 16047280 IC50 > 100000 nM T30803 CPF60C 16047281 IC50 > 100000 nM T30803 CRW35E 16047388 IC50 > 100000 nM T30803 CK8J4C 16047389 IC50 > 100000 nM T30803 C4G2DK 16048003 IC50 > 100000 nM T30803 CTLC91 16193441 IC50 > 100000 nM T30803 CZ0QS6 25269037 IC50 > 50000 nM T30803 CKM60R 25269039 IC50 > 50000 nM T30803 C1X6ZW 25269388 IC50 = 35700 nM T30803 C7ST8I 25269389 IC50 > 50000 nM T30803 C2R4CZ 25269392 IC50 > 50000 nM T30803 C97JED 25269394 IC50 > 50000 nM T30803 CH2G5I 25269395 IC50 > 50000 nM T30803 CSV31T 25269732 IC50 = 45300 nM T30803 CAO45X 25269733 IC50 > 50000 nM T30803 C6XZ7O 25269736 IC50 > 50000 nM T30803 CQ5HC3 25269737 IC50 > 50000 nM T30803 C0NL9Y 25269738 IC50 > 50000 nM T30803 C6GAR8 25269740 IC50 > 50000 nM T30803 C57MBW 25270069 IC50 > 50000 nM T30803 CN72TR 40727263 Ki = 4570 nM T30803 CCBD40 44285823 IC50 = 4000 nM T30803 CI1AD7 44286066 IC50 < 1000 nM T30803 C4U5AV 44315802 Ki > 10000000 nM T30803 CK6F2H 44322851 IC50 = 17100 nM T30803 CF9YK8 44322860 IC50 = 27200 nM T30803 CMDE38 44323177 IC50 = 13900 nM T30803 CGO0X7 44323190 IC50 = 27200 nM T30803 C2B6VO 44323235 IC50 = 9900 nM T30803 C0E4HP 44411997 IC50 > 100000 nM T30803 C7V0IZ 44412016 IC50 > 100000 nM T30803 CZ50GV 44412091 IC50 > 100000 nM T30803 CCY74J 44412123 IC50 > 100000 nM T30803 CUER27 44511333 IC50 = 6810 nM T30803 CUQB41 45266944 IC50 = 29000 nM T30803 CLGA48 45267883 IC50 = 8710 nM T30803 C3VB9U 45268767 IC50 = 23000 nM T30803 CZ3J1P 45269616 IC50 = 8100 nM T30803 CPN74S 45272169 IC50 = 10300 nM T30803 C65XIU 45273032 IC50 = 7170 nM T30803 CZ7DW4 45484008 IC50 > 50000 nM T30803 C5MB8F 46845029 IC50 = 7130 nM T30803 C60IQZ 46888469 IC50 = 11000 nM T30803 CR3Z7V 56678909 Ki = 4160 nM T30803 C83FRX 76313868 IC50 > 100000 nM T30803 C38MOW 76313869 IC50 > 100000 nM T30803 C8KR6Q 76317389 IC50 = 228000 nM T30803 C27QEH 76321111 IC50 > 100000 nM T30803 C6FC4Q 76328308 IC50 > 100000 nM T30803 C7FVU3 76331990 IC50 > 100000 nM T30803 CCX4Q3 76335573 IC50 > 100000 nM T30803 CL73RB 76335574 IC50 > 100000 nM T30803 C3B4VU 135426515 IC50 = 26700 nM T30803 C2APM1 135453064 IC50 = 7600 nM T30803 C0DGX1 135921472 IC50 > 50000 nM T30803 D03MJM 45273020 IC50 = 16000 nM T30803 D03YVX 6018993 IC50 > 100000 nM T30803 D05ABT 10352496 IC50 = 35200 nM T30803 D05CCT 4139 IC50 = 16000 nM T30803 D07TMZ 5962 Ki = 54600 nM T30803 D0A1CM 5281855 IC50 = 22800 nM T30803 D0I8HK 11665560 IC50 = 5000 nM T30803 D0L1AV 45273021 IC50 = 14200 nM T30803 D0O2DQ 237 IC50 > 1000000 nM T84703 D03ZBT 11626560 IC50 = 2 nM T84703 D04LVK 57379345 IC50 = 1829 nM T84703 D07TOK 46188928 IC50 = 5.21 nM T84703 D0AF6O 71731823 Ki = 23 nM T84703 D0OB0F 5328940 IC50 = 27 nM T84703 D00DRL 44137946 IC50 = 61 nM T84703 D01HKZ 57345941 IC50 < 3 nM T84703 D02QWY 24785538 IC50 = 4 nM T84703 D03LWG 53235510 IC50 = 3139 nM T84703 D0E3TC 44259 IC50 = 0.96 nM T84703 D0FA6S 54576299 IC50 = 4.6 nM T84703 D0FD6D 11751922 IC50 = 5 nM T84703 D0O0LS 25141092 IC50 = 3 nM T84703 D0O6WV 24794418 IC50 = 190 nM T84703 D0WS1V 448991 IC50 = 11 nM T84703 D0T3ME 156422 IC50 = 50 nM T84703 CU9J0H 2125863 IC50 = 20000 nM T84703 CY9D7W 2517470 IC50 = 20000 nM T84703 CVL95J 2535914 IC50 = 20000 nM T84703 CJ59NC 2541025 IC50 = 20000 nM T84703 C7UN1Z 2597009 IC50 = 20000 nM T84703 CF89XO 2597103 IC50 = 20000 nM T84703 CXVB08 3399504 IC50 = 20000 nM T84703 CJ3Q5R 3666186 IC50 > 10000 nM T84703 CJM9Q8 4410298 IC50 = 20000 nM T84703 CV1PK6 4798875 IC50 = 20000 nM T84703 CJU3B9 4798877 IC50 = 10461.4 nM T84703 C5AW4U 4802531 IC50 = 20000 nM T84703 CR1HA0 4802711 IC50 = 20000 nM T84703 C1DW3F 5019229 IC50 = 20000 nM T84703 CPZY43 5121984 IC50 > 50000 nM T84703 C7WO8K 7190453 IC50 = 20000 nM T84703 CDB7F4 10321590 IC50 = 646 nM T84703 CBOP58 11293798 Ki > 10000 nM T84703 C26BZX 11362471 Ki > 10000 nM T84703 CWXB93 11397177 Ki > 10000 nM T84703 CTG83F 11539329 Ki > 4500 nM T84703 CMIL86 11590363 Ki > 4500 nM T84703 C4U7HM 11621097 IC50 = 14 nM T84703 C9T6SC 11640926 Ki > 4500 nM T84703 C0AVC3 12751666 EC50 = 87.2 nM T84703 CFPW41 16007116 Ki > 4500 nM T84703 CC5J0U 16112865 IC50 = 1 nM T84703 C5VPH9 16129448 IC50 = 126 nM T84703 CFC39H 16265338 IC50 = 20000 nM T84703 C9NV2A 16272977 IC50 = 20000 nM T84703 C81LCV 16276659 IC50 = 47.1 nM T84703 C1ATH6 16322912 IC50 = 20000 nM T84703 C2HVS1 16739794 IC50 < 1 nM T84703 C03EXR 16739855 IC50 = 1 nM T84703 CW64AB 16739883 IC50 = 1 nM T84703 CD7B6L 17561456 IC50 = 20000 nM T84703 CE1TZ9 20971557 IC50 = 20000 nM T84703 CQHK69 23646624 IC50 = 160 nM T84703 CJ0CU5 24825841 IC50 = 9.37 nM T84703 CY8L7E 24896769 IC50 > 10000 nM T84703 C0KMW8 24937716 IC50 = 13 nM T84703 C5WG1H 24937847 IC50 = 11 nM T84703 C8CO4B 24971342 IC50 = 1100 nM T84703 C3DI7Y 24995523 IC50 = 5 nM T84703 C76PSW 44518384 IC50 = 50 nM T84703 C6LP9V 44518674 IC50 = 47 nM T84703 C36KYB 44520611 IC50 = 29 nM T84703 CZH80Q 44520612 IC50 = 1970 nM T84703 CY3HW5 46224684 IC50 > 10000 nM T84703 CBI7V6 46382265 IC50 = 20000 nM T84703 CMP5T4 46382269 IC50 = 20000 nM T84703 CRP7H0 46382271 IC50 = 5460.3 nM T84703 CT5ZD0 46382272 IC50 = 9064.5 nM T84703 COB29T 46382277 IC50 = 20000 nM T84703 C7TY0M 46382278 IC50 = 20000 nM T84703 CUCX57 46382281 IC50 = 20000 nM T84703 CGR3T6 46382286 IC50 = 20000 nM T84703 CPZ81K 46382288 IC50 = 20000 nM T84703 CU9IK7 46382290 IC50 = 20000 nM T84703 C61WCT 46382295 IC50 = 20000 nM T84703 C4P1AT 46382302 IC50 = 3224.9 nM T84703 CMDC48 46382303 IC50 = 20000 nM T84703 C2ZA3E 46382304 IC50 = 1196.8 nM T84703 CN5R0P 46382305 IC50 = 20000 nM T84703 CH53ZD 46382308 IC50 = 20000 nM T84703 CT3UO5 46382309 IC50 = 20000 nM T84703 C3R5DF 46382310 IC50 = 20000 nM T84703 CVP36M 46382311 IC50 = 20000 nM T84703 CEP0C1 46382312 IC50 = 20000 nM T84703 CUG2W7 46382314 IC50 = 423.2 nM T84703 CDOR02 46382315 IC50 = 2594.4 nM T84703 CG6D4E 46382317 IC50 = 2843.4 nM T84703 C2L3WY 46382318 IC50 = 20000 nM T84703 CPA41J 46382319 IC50 = 20000 nM T84703 C54EDX 46382322 IC50 = 20000 nM T84703 C9J1CQ 46382323 IC50 = 20000 nM T84703 C37VDC 46382324 IC50 = 778 nM T84703 CG13SB 46382326 IC50 = 20000 nM T84703 CD3QY0 46382327 IC50 = 20000 nM T84703 C6ZNO1 46382331 IC50 = 20000 nM T84703 CE6N3J 46382332 IC50 = 20000 nM T84703 COD4I0 46382336 IC50 = 20000 nM T84703 CGD5Q0 46382338 IC50 = 20000 nM T84703 C40NSR 46382339 IC50 = 20000 nM T84703 C8H2CR 46382341 IC50 = 20000 nM T84703 C64RBV 46382343 IC50 = 20000 nM T84703 C6NS1L 46382344 IC50 = 20000 nM T84703 CP23VF 46382346 IC50 = 20000 nM T84703 CP9W3T 46382349 IC50 = 20000 nM T84703 CZNH36 46382354 IC50 = 3886.6 nM T84703 CYH93R 46382355 IC50 = 3575.6 nM T84703 CV51XI 46382356 IC50 = 20000 nM T84703 C7SKH2 46382366 IC50 = 20000 nM T84703 CJD49N 46382375 IC50 = 20000 nM T84703 CJ8E1N 46382394 IC50 = 20000 nM T84703 CW4EI1 46390524 IC50 = 20000 nM T84703 CQG51S 46390527 IC50 = 20000 nM T84703 CZ49OG 46390528 IC50 = 20000 nM T84703 CSJ20W 46390529 IC50 = 10000 nM T84703 CRAK47 46390532 IC50 = 20000 nM T84703 CLS29B 46872626 IC50 > 10000 nM T84703 C2O8RZ 46886323 IC50 > 1000 nM T84703 C1NKE3 46905987 IC50 > 3000 nM T84703 C8KT1S 50802118 IC50 = 20000 nM T84703 C2X9OA 50802180 IC50 = 20000 nM T84703 CF57GW 50802181 IC50 = 2138.5 nM T84703 C1ED3N 50802184 IC50 = 10000 nM T84703 C6G1LV 50802187 IC50 = 20000 nM T84703 CC3YE6 50802196 IC50 = 10000 nM T84703 CBF28N 50802197 IC50 = 20000 nM T84703 CK6G9M 50802198 IC50 = 771 nM T84703 CIC1B4 50802201 IC50 = 9280 nM T84703 CWCP03 50802214 IC50 = 10000 nM T84703 CQP98F 50802215 IC50 = 2497.3 nM T84703 CVT2O0 50802216 IC50 = 10000 nM T84703 C2G4HZ 50802217 IC50 = 10000 nM T84703 CB1AM0 50802226 IC50 = 20000 nM T84703 CNRX75 50802227 IC50 = 10000 nM T84703 COJ6T7 50802228 IC50 = 20000 nM T84703 CH4K8I 50802229 IC50 = 10000 nM T84703 CST50B 50802232 IC50 = 10000 nM T84703 CI9H3K 50802245 IC50 = 20000 nM T84703 C1LHW9 50802246 IC50 = 20000 nM T84703 C7IQV2 50802247 IC50 = 20000 nM T84703 CY61RH 50802250 IC50 = 10000 nM T84703 CEA48B 50802259 IC50 = 20000 nM T84703 CRT9S8 50802262 IC50 = 4615.5 nM T84703 C23SQR 50802263 IC50 = 20000 nM T84703 C5IZR7 50802274 IC50 = 9792.4 nM T84703 CVR8K4 50802276 IC50 = 10000 nM T84703 C4WMI1 50802277 IC50 = 20000 nM T84703 CG52PC 50802293 IC50 = 20000 nM T84703 CQ3R5U 50802295 IC50 = 20000 nM T84703 CB3CE4 50802298 IC50 = 2027.5 nM T84703 C3FYU7 50802299 IC50 = 20000 nM T84703 C8A6MI 50802307 IC50 = 20000 nM T84703 C94SOF 50802309 IC50 = 63.7 nM T84703 C4Y6SN 50802310 IC50 = 358.6 nM T84703 CCKR79 50802312 IC50 = 10000 nM T84703 CFA79B 50802314 IC50 = 20000 nM T84703 CB8PD0 50802328 IC50 = 10000 nM T84703 C17YAG 50802329 IC50 = 6706 nM T84703 CSL61K 50802332 IC50 = 20000 nM T84703 CGBH51 50802345 IC50 = 10000 nM T84703 C13KBR 50802348 IC50 = 10000 nM T84703 C5SZE1 50802358 IC50 = 10000 nM T84703 C0F1XK 50802359 IC50 = 20000 nM T84703 CE4HR6 50802360 IC50 = 20000 nM T84703 CU5B4V 50802364 IC50 = 20000 nM T84703 CV9PN1 50802374 IC50 = 1340.8 nM T84703 C17PKR 50802391 IC50 = 20000 nM T84703 CJ7G2O 50802392 IC50 = 10000 nM T84703 C5V3JC 50802393 IC50 = 10000 nM T84703 C8JKA9 50802404 IC50 = 20000 nM T84703 C16UZW 50802409 IC50 = 20000 nM T84703 C7KC5M 50802410 IC50 = 20000 nM T84703 CX7BU6 50802411 IC50 = 10000 nM T84703 C5RI6H 50802419 IC50 = 10000 nM T84703 CR6GC8 50802420 IC50 = 10000 nM T84703 C6R1VG 50802424 IC50 = 10000 nM T84703 C6O9GD 50802433 IC50 = 20000 nM T84703 C9UR2X 50825254 IC50 = 20000 nM T84703 CWR12L 50825338 IC50 = 20000 nM T84703 CH6OS5 50825345 IC50 = 20000 nM T84703 CVYM85 50825346 IC50 = 20000 nM T84703 CM24LF 52938983 IC50 < 1 nM T84703 C8NA4L 53384644 IC50 = 8700 nM T84703 C6U0SG 57629460 IC50 = 1 nM T84703 C1EVX0 58063117 IC50 = 5380 nM T84703 CSG5T1 58335664 IC50 = 4 nM T84703 C0HR7L 59804298 IC50 = 27 nM T84703 CZM10S 59804305 IC50 = 15 nM T84703 CJ1BN7 59804319 IC50 = 7 nM T84703 CUQ6Y0 59804322 IC50 = 60 nM T84703 C8ZF3L 59804374 IC50 = 35 nM T84703 C37NKO 67129970 IC50 = 5240 nM T84703 CK80LJ 67130050 IC50 > 10000 nM T84703 CV63UL 67240318 IC50 > 10000 nM T84703 C0VJW8 68545858 IC50 = 21 nM T84703 C7GRV2 68755406 IC50 = 8340 nM T84703 C7VJ6A 70647728 IC50 = 100 nM T84703 C3PX5C 70692373 IC50 = 17 nM T84703 CXZ40O 70696497 IC50 = 19 nM T84703 CKT60L 71455860 Ki > 4500 nM T84703 CRI51K 73819548 Ki = 0.4 nM T84703 CGDB30 74538658 IC50 = 190 nM T84703 CIQ5D8 74627727 IC50 = 132.2 nM T84703 CRSY98 89808125 Ki = 77 nM T84703 C40VNJ 89816720 Ki = 65 nM T84703 CM64AB 90644193 Ki = 0.5 nM T84703 CI4N8P 91801232 IC50 = 0.3 nM T84703 CLZ74S 91826737 IC50 = 94000 nM T84703 CJQ5N6 91936970 IC50 = 1190000 nM T84703 C3PAN1 117967296 IC50 > 81000 nM T84703 CE86QC 118128728 IC50 = 1303.7 nM T84703 C0TMZ8 118167692 IC50 = 2.6 nM T84703 CLH8X7 118189551 IC50 = 6.1 nM T84703 CU3K0B 118456253 IC50 = 14000 nM T84703 C60TWO 118665627 IC50 = 15 nM T84703 CPK47S 118868365 IC50 = 6.2 nM T84703 CN4X0C 121231414 IC50 = 36.8 nM T84703 C08KEM 122179540 IC50 = 270 nM T84703 CQ43XF 122179541 IC50 = 200 nM T84703 C2TXZ9 122179542 IC50 = 120 nM T84703 CXS1Y6 122179543 IC50 = 27 nM T84703 CPF2L7 122179544 IC50 = 7 nM T84703 C3NJ6T 122179545 IC50 = 130 nM T84703 C3AJ4C 122179546 IC50 = 1 nM T84703 CG0RP7 122179547 IC50 = 1 nM T84703 C1A0SQ 122179548 IC50 = 4 nM T84703 C4X7SD 122192466 IC50 > 10000 nM T84703 CC83HO 123131777 IC50 = 27000 nM T84703 C93UNX 132041675 IC50 = 4.2 nM T84703 C1X6FJ 134693894 IC50 = 40 nM T84703 CXC69T 137321158 IC50 = 8 nM T84703 CWC49K 137321210 IC50 > 1000 nM T84703 CI1E8V 137634241 IC50 = 379 nM T84703 CNRT47 139434032 EC50 = 790 nM T84703 CIN6L7 139434035 EC50 = 370 nM T84703 CTFE03 139434036 EC50 = 230 nM T84703 CX9H4W 139434047 EC50 = 750 nM T84703 CU10QZ 139434077 EC50 = 370 nM T84703 CLRW84 139434103 EC50 = 950 nM T84703 CB6F5R 139434105 EC50 = 1400 nM T84703 C7FBY1 139434107 EC50 = 390 nM T84703 C08MUD 139434127 EC50 = 250 nM T84703 C2MZ4L 139434198 EC50 = 610 nM T84703 CJIH42 139434200 EC50 = 270 nM T84703 C7W5MH 139434224 EC50 = 110 nM T84703 CXIT16 139434239 EC50 = 460 nM T84703 C2B8OV 139442846 EC50 = 120 nM T84703 C4ID6F 139442949 EC50 = 450 nM T84703 CX4E3H 142736778 IC50 = 4.42 nM T84703 CAJQ14 145964002 IC50 = 6.6 nM T84703 CVF4M6 145965985 IC50 = 2.7 nM T84703 C5MHK6 145967970 IC50 = 900 nM T84703 CK9C0H 145970062 IC50 = 29 nM T84703 CI85EU 145998085 IC50 > 1000 nM T84703 CA10CQ 155512867 IC50 > 1000 nM T84703 C2MD1Q 155513187 IC50 > 10000 nM T84703 C5B2AX 155513312 IC50 = 24.19 nM T84703 CZMD64 155514443 IC50 > 1000 nM T84703 CB5T9G 155515436 IC50 = 145.4 nM T84703 CUHZ87 155516883 IC50 > 1000 nM T84703 COR4M0 155517181 IC50 = 20000 nM T84703 CIU1T6 155518465 IC50 = 41.34 nM T84703 C86HPW 155518524 IC50 = 6300 nM T84703 CO63MP 155519543 IC50 = 10.47 nM T84703 C9TU2A 155520832 IC50 = 5000 nM T84703 CBG4P0 155524103 IC50 = 43.47 nM T84703 CN6C2T 155528463 IC50 = 13.11 nM T84703 C0HW7F 155530527 IC50 > 1000 nM T84703 CP5IW9 155530600 IC50 > 1000 nM T84703 C3MC2P 155532434 IC50 = 178.45 nM T84703 CNE6A3 155532801 IC50 = 38.35 nM T84703 C2KAU0 155533663 IC50 = 22.73 nM T84703 C75AKY 155533695 IC50 < 10 nM T84703 C3PWI1 155534046 IC50 > 1000 nM T84703 CTXK93 155535665 IC50 = 270.7 nM T84703 C14SEB 155535950 IC50 = 343.9 nM T84703 CV9D5J 155536164 IC50 = 315.13 nM T84703 C3O6WX 155540330 IC50 > 1000 nM T84703 C76NKG 155543431 IC50 > 1000 nM T84703 CRV40J 155546026 IC50 = 253.65 nM T84703 C8AG4U 155550655 IC50 = 15.59 nM T84703 C2RQT8 155550913 IC50 < 10 nM T84703 C9MJL5 155551408 IC50 > 1000 nM T84703 CM7Q3F 155556300 IC50 = 1500 nM T84703 C9OLA3 155557330 IC50 = 0.2 nM T84703 CYD1C7 155560599 IC50 > 1000 nM T84703 C40IYS 155562258 IC50 = 58.8 nM T84703 CBG9Z1 155562952 IC50 = 569 nM T84703 C0WZ9S 155563842 IC50 > 1000 nM T84703 CWR4O5 155565233 IC50 = 9.3 nM T84703 CRFW02 155566430 IC50 = 43.92 nM T84703 C0V7SM 155567015 IC50 > 1000 nM T84703 D00ERW 44444843 Ki > 4536 nM T84703 D00HVA 11624601 Ki > 4500 nM T84703 D02RWC 59397065 IC50 = 12 nM T84703 D07ADX 54764565 IC50 = 217 nM T84703 D0E7VO 59627005 IC50 < 100 nM T84703 D0K5UF 72710568 IC50 = 4 nM T84703 D0L3JR 25212148 IC50 = 9 nM T84703 D0N4LR 53469448 IC50 = 2962 nM T84703 D0O8AR 16097523 IC50 = 0.93 nM T84703 D0Q3NG 11715520 Ki > 4500 nM T84703 D0R2WK 16038120 IC50 = 2018 nM T84703 D0S7IE 11658882 Ki > 4500 nM T89697 D00AXJ 4189 IC50 = 1400 nM T89697 D03GET 4055 IC50 = 370 nM T89697 D04GYO 5353853 IC50 = 28000 nM T89697 D05EJG 6305 IC50 = 498700 nM T89697 D0AA2D 2378 IC50 = 23000 nM T89697 D0EV8E 3198 IC50 = 1100 nM T89697 D0O6UZ 65863 IC50 = 8400 nM T89697 D0P9AC 3675 IC50 = 14000 nM T89697 D0X8XA 5318 IC50 = 6400 nM T89697 D0Y0GH 5746 Ki = 25000 nM T89697 D06MHZ 66558287 Ki = 7 nM T89697 D08CJK 1150 Ki = 156000 nM T89697 D0B1FE 3194 Ki = 94 nM T89697 D0B5HS 405012 EC50 = 110000 nM T89697 D0C0NH 3806 IC50 = 1000 nM T89697 D0DA5M 75202656 IC50 = 23 nM T89697 D0DP5I 121328278 IC50 = 0.5 nM T89697 D0J1HB 23063810 IC50 = 410 nM T89697 D0PM5U 135564890 IC50 = 7 nM T89697 D0W0VD 3885 Ki = 100 nM T89697 D09HVV 118898844 IC50 = 3 nM T89697 D0MQ3X 5316743 IC50 = 1300 nM T89697 D0QZ8K 70874141 EC50 = 330 nM T89697 D0S7BW 78426054 IC50 < 1000 nM T89697 D0WR7B 122650373 IC50 = 9.7 nM T89697 D0YY4R 121339537 IC50 = 3 nM T89697 D0R7MJ 135403797 IC50 = 60000 nM T89697 C6A3UH 3037 IC50 = 70000 nM T89697 C0RFA2 3102 IC50 = 1000000 nM T89697 C9LCD8 3823 IC50 = 25000 nM T89697 CP62OB 5138 IC50 = 61000 nM T89697 CXHL15 6755 IC50 = 675000 nM T89697 C2JK3W 7104 IC50 = 1000000 nM T89697 COE28J 7220 IC50 = 2570000 nM T89697 CEUJ71 7400 IC50 > 20000 nM T89697 CV9D7A 7516 IC50 = 230 nM T89697 C9KP5F 7518 IC50 = 9200 nM T89697 CV79ZO 7564 IC50 = 400000 nM T89697 CJ19CF 7812 IC50 = 1319000 nM T89697 C45VRP 7815 IC50 = 1900 nM T89697 CM75BH 8447 IC50 > 500000 nM T89697 CG47UK 10241 IC50 > 200000 nM T89697 CBIR94 10313 IC50 = 16000 nM T89697 COI9A4 10852 IC50 = 61000 nM T89697 C25MFK 11157 IC50 = 71000 nM T89697 COZB91 11988 IC50 = 8000 nM T89697 C08ZTB 13397 IC50 > 20000 nM T89697 CGC0N1 13886 IC50 = 161000 nM T89697 CE4X3M 21095 IC50 = 3970 nM T89697 CUP89L 22244 IC50 = 15000 nM T89697 C0HZ4G 22641 IC50 = 1000000 nM T89697 CC0BW7 22704 IC50 > 500000 nM T89697 CA90DS 23116 IC50 = 800 nM T89697 COY1P0 32238 IC50 = 130000 nM T89697 CL1A5R 37175 IC50 = 23000 nM T89697 C51XBL 40302 IC50 = 1000000 nM T89697 C2HMI7 66036 IC50 > 20000 nM T89697 C0F5BM 67430 IC50 > 20000 nM T89697 C1B9ZO 68094 IC50 = 2000000 nM T89697 C3AVU2 72732 IC50 = 4340 nM T89697 CW95YM 73468 IC50 = 22600 nM T89697 C1BI4N 74318 IC50 > 1000000 nM T89697 CYH1I4 74787 IC50 = 870 nM T89697 CHO9A0 74967 IC50 = 2700 nM T89697 CDL20X 75899 IC50 > 1000000 nM T89697 CRY89S 83050 IC50 = 500000 nM T89697 CSMK07 98112 IC50 = 14690 nM T89697 CB4VI8 99128 IC50 = 114000 nM T89697 C3CKU4 102313 IC50 < 10000 nM T89697 CD68XC 104251 IC50 = 400000 nM T89697 CD24AO 114918 Ki = 326 nM T89697 CBZX05 120425 IC50 = 24000 nM T89697 CS53VH 128994 IC50 = 4680 nM T89697 C5LQN0 199162 IC50 = 10000 nM T89697 CTDZ45 201863 EC50 = 2000 nM T89697 CUG38M 203812 IC50 = 410 nM T89697 CH0ZD7 207299 IC50 = 134 nM T89697 CN6O1K 217573 IC50 = 1300 nM T89697 CNQE70 224502 IC50 = 21000 nM T89697 CCQ3W7 233294 IC50 = 35600 nM T89697 C8PEY0 234811 IC50 = 400 nM T89697 CR36LZ 235240 Ki > 100000 nM T89697 CFPL09 236715 IC50 = 1780 nM T89697 CR48HG 239465 IC50 = 750 nM T89697 C37KML 244989 IC50 = 15700 nM T89697 CVO36F 248768 IC50 = 6300 nM T89697 C4MLK5 255448 IC50 = 1600 nM T89697 CRJ5W7 259418 IC50 = 1500 nM T89697 CU3D0T 261066 IC50 = 42500 nM T89697 CR1C6K 261602 IC50 = 714 nM T89697 CE7M6K 269624 Ki = 4300 nM T89697 CLC05O 272989 IC50 = 1950 nM T89697 CRF3E1 273059 IC50 = 8200 nM T89697 CR9VJ4 273769 IC50 = 332 nM T89697 CS46CV 276137 IC50 = 35600 nM T89697 CY3BT7 291128 IC50 = 31600 nM T89697 CV57WU 291217 IC50 = 266000 nM T89697 C9TU7X 291363 IC50 = 32600 nM T89697 C8GDA3 302654 IC50 = 44900 nM T89697 C1OA7G 313613 IC50 = 3300 nM T89697 C0UAT7 313614 IC50 = 660 nM T89697 C8RHI3 313619 IC50 = 24000 nM T89697 CJ1V4S 325901 IC50 = 42500 nM T89697 CC2M9A 332650 IC50 = 4100 nM T89697 C4HP3I 332972 IC50 = 4900 nM T89697 COK78A 333769 IC50 = 6080 nM T89697 C3RMI4 333770 IC50 = 34960 nM T89697 C8BS0X 334304 IC50 = 464000 nM T89697 CA1H8B 336270 IC50 = 183 nM T89697 CL2JH7 336699 IC50 = 930 nM T89697 CD3RI9 356301 IC50 = 76000 nM T89697 CDK1S3 356303 IC50 = 96000 nM T89697 CM49EY 362360 IC50 = 460 nM T89697 CVD5W0 363326 IC50 = 3000 nM T89697 C7EZ4T 369539 IC50 = 1000000 nM T89697 CNS32X 371271 IC50 = 35600 nM T89697 CUR85O 378581 IC50 = 46700 nM T89697 CB9RU8 421540 IC50 > 10000 nM T89697 CQ7P3K 432556 IC50 = 890 nM T89697 C46VHU 478572 IC50 = 53.9 nM T89697 C72ZLN 478574 IC50 = 23 nM T89697 CC7IW3 478577 IC50 = 121200 nM T89697 C2ZR8M 478643 IC50 = 466 nM T89697 CY38AJ 478645 IC50 = 864400 nM T89697 CZT01E 478647 IC50 = 27.1 nM T89697 CD1AO0 487082 IC50 = 4400 nM T89697 C74FPR 497025 Ki = 35 nM T89697 C03NZX 523214 IC50 = 156 nM T89697 C4ONK2 555630 IC50 = 490 nM T89697 CR2L7A 600260 IC50 = 6000000 nM T89697 CZI5R2 601577 IC50 = 817000 nM T89697 CN7WA6 615185 IC50 = 4800 nM T89697 CD3V5T 651817 IC50 > 100000 nM T89697 C8K5LQ 657876 IC50 = 123000 nM T89697 C6C9AZ 658687 IC50 = 50000 nM T89697 CEM8K0 685364 IC50 = 195000 nM T89697 C6NX0C 689063 IC50 = 90490 nM T89697 CKMP38 697993 IC50 = 126000 nM T89697 C7M4VB 698285 IC50 = 1800 nM T89697 CO46LB 706988 IC50 > 50000 nM T89697 CNV69W 707050 IC50 = 15000 nM T89697 C5W2PB 717704 IC50 > 50000 nM T89697 CV53ZJ 725906 IC50 = 1690 nM T89697 C6WQ0V 735843 IC50 > 20000 nM T89697 CM7C6Y 737132 IC50 > 50000 nM T89697 C3WG8U 737138 IC50 > 50000 nM T89697 C5LN3R 737149 IC50 = 1800 nM T89697 CUMJ16 737276 IC50 > 50000 nM T89697 CO5F6Z 737504 IC50 = 41000 nM T89697 CAG2B4 763555 IC50 = 522000 nM T89697 CK89WR 781705 IC50 = 112000 nM T89697 CY02AP 795453 IC50 = 71 nM T89697 CI43WJ 802727 IC50 = 1800 nM T89697 CG54RM 802728 IC50 = 83000 nM T89697 C64NSF 819511 IC50 = 35000 nM T89697 CDEF92 820765 IC50 = 5888.44 nM T89697 CXYV26 849731 IC50 = 767 nM T89697 C47XAO 849732 IC50 > 10000 nM T89697 CB27WS 849733 IC50 = 808.9 nM T89697 C5S9DF 849734 IC50 = 4612 nM T89697 C34QEU 849735 IC50 = 1770 nM T89697 CC10TB 852498 IC50 = 65000 nM T89697 CFD05W 992980 IC50 = 20100 nM T89697 C85BIS 992984 IC50 = 3200 nM T89697 CXWM34 993112 IC50 = 5600 nM T89697 CEQ35N 1016842 IC50 = 18000 nM T89697 CSC0B6 1041635 IC50 = 2587 nM T89697 CY6C8D 1085103 IC50 = 1190 nM T89697 CK4G6F 1167203 IC50 = 12400 nM T89697 CT2F4J 1479909 IC50 = 2600 nM T89697 CTE7D4 1484508 IC50 > 20000 nM T89697 C7NOW6 1712812 IC50 = 82000 nM T89697 C5D0MU 1810299 IC50 > 50000 nM T89697 C25ERJ 1810302 IC50 = 17000 nM T89697 C4QW9C 2728703 IC50 = 1000 nM T89697 CI85YE 2731263 IC50 > 50000 nM T89697 C0FH4G 2732070 IC50 > 20000 nM T89697 CY78SE 2735617 IC50 = 1600 nM T89697 CN35FD 2737499 IC50 = 3700 nM T89697 C7I1HC 2744597 IC50 = 38610 nM T89697 C94BMC 2757941 IC50 > 50000 nM T89697 C3IRL6 2758211 IC50 = 18000 nM T89697 CQ6Z8A 2759372 IC50 = 3500 nM T89697 CYD7A1 2764014 IC50 = 630 nM T89697 CHS3B0 2794173 IC50 = 6000 nM T89697 C84XTS 2803091 IC50 = 11700 nM T89697 CHJQ46 2806436 IC50 = 6300 nM T89697 CXM75A 2807416 IC50 = 3100 nM T89697 CCEN29 2810177 IC50 = 13000 nM T89697 C59BGS 2818222 IC50 > 100000 nM T89697 C1H3JC 2821620 IC50 = 97000 nM T89697 CN7MC6 2821621 IC50 = 15000 nM T89697 CHB3S4 2821626 IC50 = 4600 nM T89697 CK2FZ7 2821627 IC50 = 18000 nM T89697 CG8L6W 2824871 IC50 = 710 nM T89697 CM9J0C 2825091 IC50 = 2000000 nM T89697 C7X5WE 2828334 IC50 = 110 nM T89697 CU6Z9O 2917429 Ki = 342300 nM T89697 C3KZ0U 3028808 IC50 = 2000 nM T89697 CHRQ07 3032509 Ki = 72410 nM T89697 C09JXD 3032646 Ki = 62360 nM T89697 C37ABE 3035211 Ki = 12000 nM T89697 C6ZP2C 3106159 IC50 = 1000 nM T89697 C7D6IH 3161266 IC50 = 310000 nM T89697 C53LIN 3325609 EC50 = 128 nM T89697 C61GRB 3443692 IC50 = 2400 nM T89697 CZ9IS6 3529520 IC50 = 120 nM T89697 CB0D8U 3595344 EC50 = 3118 nM T89697 C7O9DU 3720080 IC50 = 2600 nM T89697 CIO57N 3761458 IC50 > 20000 nM T89697 C12IDC 3901929 IC50 = 1510 nM T89697 C7DM2Y 4099901 IC50 = 108000 nM T89697 CV10YZ 4190125 EC50 = 420 nM T89697 CA3PO5 4240303 EC50 > 10 nM T89697 CH6K0A 4310362 IC50 = 68000 nM T89697 C87WUF 4381769 IC50 = 15000 nM T89697 CNUQ02 4456830 IC50 = 1580 nM T89697 CB5P9D 4574587 IC50 = 379.5 nM T89697 C45WVE 4638522 EC50 = 640 nM T89697 CZNE04 4794706 IC50 = 49 nM T89697 CU6XY2 5068606 IC50 = 26000 nM T89697 C0VGT3 5170924 IC50 > 50000 nM T89697 CAW37X 5240714 IC50 = 3740 nM T89697 C8KM3N 5371761 IC50 = 110 nM T89697 CS67OL 5712754 IC50 = 20000 nM T89697 C9C5OF 5937842 IC50 = 50000 nM T89697 CFGA74 6198019 Ki = 3000 nM T89697 C1RPA8 6223130 EC50 = 13260 nM T89697 CL82TX 6400901 IC50 = 940 nM T89697 CGP9S8 6409664 IC50 = 620 nM T89697 C3AV5I 6419227 IC50 = 22000 nM T89697 CIQ4X3 6419341 IC50 = 1256000 nM T89697 C5KX9O 6494204 Ki = 35 nM T89697 CXE93M 6494205 Ki = 35 nM T89697 CP1O4X 7064051 IC50 = 2700 nM T89697 CR0P9A 7463552 IC50 = 17910 nM T89697 CN16IB 8005342 EC50 = 609 nM T89697 CP61HD 8070877 IC50 = 9750 nM T89697 CZ06FE 8071109 IC50 = 30800 nM T89697 CN9Y1O 8106455 IC50 > 100000 nM T89697 CP43WG 8106458 IC50 > 20000 nM T89697 CNW5G7 9573924 Ki = 1500 nM T89697 C0PE9C 9584160 IC50 = 60000 nM T89697 C7HIG1 9584719 IC50 = 31000 nM T89697 C8VKT5 9685191 IC50 = 2780 nM T89697 CAVT12 9812842 IC50 = 39000 nM T89697 C4UYP5 9815283 IC50 > 100000 nM T89697 CQ25OP 9833992 IC50 = 680000 nM T89697 C4QZ1I 9877471 IC50 = 190000 nM T89697 C7N9PW 9877511 IC50 = 1028000 nM T89697 C71STY 9899224 IC50 = 2300000 nM T89697 C6NS2U 9899225 IC50 = 6000 nM T89697 CU3RN8 9920462 IC50 = 70000 nM T89697 C69CDF 9920916 IC50 = 2600 nM T89697 C2PCN3 9964175 IC50 = 1500000 nM T89697 CUP4N1 9964258 Ki = 14500 nM T89697 CE64VW 10101379 IC50 = 440 nM T89697 CQC7N5 10332864 IC50 = 80.3 nM T89697 C4XB1O 10355804 IC50 = 140000 nM T89697 CH8N5K 10374898 IC50 = 190000 nM T89697 CYO69B 10511388 IC50 = 825000 nM T89697 C9JU5L 10559053 IC50 = 41000 nM T89697 CL21AV 10583021 IC50 = 5700 nM T89697 C8GMF7 10890197 IC50 > 100000 nM T89697 C7Q6NX 10909696 IC50 = 1800000 nM T89697 CI3T6M 11086357 IC50 = 4950 nM T89697 CYKR73 11175492 Ki = 35 nM T89697 CFD24O 11209246 Ki = 35 nM T89697 C4RKW2 11255489 Ki = 35 nM T89697 C32WXK 11275256 IC50 = 2900 nM T89697 CB50ZE 11423685 IC50 = 422000 nM T89697 C2P0LW 11482022 Ki = 47570 nM T89697 CJ3AO4 11528610 Ki = 1292000 nM T89697 C9A3BN 11528678 Ki = 42060 nM T89697 C5AI2W 11536281 Ki = 33970 nM T89697 CGT35V 11543253 Ki = 179600 nM T89697 CF5C4D 11580169 IC50 = 420 nM T89697 C5H7ZN 11629967 Ki = 1267000 nM T89697 CL48GN 11651542 Ki = 149350 nM T89697 CZS94C 11673059 Ki = 328700 nM T89697 CZS6U0 11694196 IC50 = 650000 nM T89697 CXKY79 11701328 Ki = 202000 nM T89697 CEM3R0 11708775 Ki = 40950 nM T89697 CT7KH0 11757335 IC50 = 15000 nM T89697 C4Q1MV 12014591 Ki = 35 nM T89697 CD6L1H 12239941 IC50 = 2920 nM T89697 CQ9ZI8 12239942 IC50 = 121 nM T89697 C53LFZ 12240982 IC50 = 533000 nM T89697 CQN15E 12243104 IC50 = 22000 nM T89697 C1MS3C 12244898 IC50 = 61000 nM T89697 CT0AG4 12398786 IC50 > 20000 nM T89697 CW0OD3 12398789 IC50 > 100000 nM T89697 CSM6Z7 12457713 IC50 > 50000 nM T89697 C3NTB9 12463137 IC50 = 1200000 nM T89697 CYO6J1 12471537 IC50 = 460000 nM T89697 C1FL0I 12474093 IC50 = 3400 nM T89697 CRX8P7 12674978 IC50 = 1970 nM T89697 C9BJU0 12722498 IC50 > 50000 nM T89697 C5PD2B 12760607 IC50 = 200000 nM T89697 C29LGR 12800721 IC50 = 980 nM T89697 C39AWQ 13393248 IC50 = 3390 nM T89697 CQ21YE 13762869 IC50 = 779 nM T89697 C3Y2XJ 14034883 IC50 = 190 nM T89697 CC94WU 14171303 IC50 = 29 nM T89697 CYE1A6 14171304 IC50 = 26.2 nM T89697 CW53FC 14269350 IC50 = 24920 nM T89697 C19VME 14269353 IC50 = 50810 nM T89697 C7G0ME 14269354 IC50 = 62660 nM T89697 CO2TC8 14694516 IC50 = 18000 nM T89697 C96HAY 14736077 IC50 > 20000 nM T89697 C7XD2T 15118768 Ki = 635000 nM T89697 C9MNU7 15326268 IC50 = 370 nM T89697 CTF31B 15326270 IC50 = 53000 nM T89697 C83DSK 15754003 IC50 = 13000 nM T89697 CXW9D2 15946462 Ki = 210 nM T89697 C0W9ID 16059788 Ki = 120 nM T89697 CMJV13 16069892 IC50 > 30000 nM T89697 C07KDO 16069930 IC50 > 30000 nM T89697 C3J1EB 16069933 IC50 = 20600 nM T89697 CM74CV 16069934 IC50 > 30000 nM T89697 CKH6M4 16090079 IC50 = 977 nM T89697 CQ7B2J 16118954 Ki = 82540 nM T89697 CGDT43 16228806 IC50 = 1500 nM T89697 C91JFG 17750145 IC50 = 320 nM T89697 CNR81H 17995458 IC50 = 1000000 nM T89697 CB21MY 18314043 IC50 > 20000 nM T89697 CNS59Y 18506325 IC50 = 1028000 nM T89697 CTS6O0 18525978 IC50 = 1600 nM T89697 C2IQL8 18525980 IC50 = 450 nM T89697 C68SNL 18525982 IC50 = 2500 nM T89697 CAF4Q6 18525983 IC50 = 5400 nM T89697 C3C7JL 18525997 IC50 = 9500 nM T89697 CZ84SF 18526040 IC50 = 8900 nM T89697 CS84LJ 19702149 IC50 = 60000 nM T89697 CEL18N 19974989 IC50 = 630 nM T89697 CQIY45 20373984 IC50 = 209000 nM T89697 C2ID7K 20525178 IC50 = 830000 nM T89697 C2B0PJ 21125239 IC50 = 340 nM T89697 C4EOJ3 21155916 IC50 = 880 nM T89697 CP37KN 21192890 IC50 = 1400 nM T89697 C0VLB8 21683122 IC50 = 2100 nM T89697 C08CBI 21723626 IC50 = 24000 nM T89697 C50TDQ 21798789 IC50 = 820000 nM T89697 CGM9O7 22009901 IC50 > 100000 nM T89697 C4J1QN 22989754 IC50 = 7100 nM T89697 C1BI5L 22989786 IC50 = 1680 nM T89697 C07TJG 22989894 IC50 = 12000 nM T89697 CEM41C 23063802 IC50 = 830 nM T89697 C0TJ5U 23084904 IC50 = 179000 nM T89697 C0CIY4 23084917 IC50 = 60000 nM T89697 CPC8I6 23206139 IC50 = 1000 nM T89697 CQ93UJ 23332019 IC50 = 1300000 nM T89697 C3P4TR 23766450 Ki = 35 nM T89697 C3BVO4 24264313 IC50 > 100000 nM T89697 CBXC05 24424330 IC50 = 37000 nM T89697 C0Z3PM 24741909 IC50 = 2310 nM T89697 CP4I3W 24742062 IC50 = 94000 nM T89697 CSK1I0 24788785 Ki = 260 nM T89697 CQ16CP 24822271 IC50 = 247 nM T89697 CZ5PI3 24822272 IC50 = 5520 nM T89697 C4BOC3 24822273 IC50 = 2050 nM T89697 C40EMQ 24824456 IC50 = 2130 nM T89697 CAL06M 24824607 IC50 = 3020 nM T89697 C1JN8S 24824608 IC50 = 933 nM T89697 CPFN24 24824612 IC50 = 130 nM T89697 CWO6G7 24825243 Ki = 41 nM T89697 CO29PG 24825244 Ki = 1490 nM T89697 CF65SE 24825245 Ki = 10900 nM T89697 C4HY5W 24825246 Ki = 420 nM T89697 C3PE8G 24825247 Ki = 200 nM T89697 CJ5O3I 24825249 Ki = 260 nM T89697 C9TH2J 24971328 Ki = 4800 nM T89697 C4OA9Q 24971329 IC50 = 25000 nM T89697 C7FWD4 24971330 IC50 = 38000 nM T89697 CV1IW8 24971331 IC50 = 73000 nM T89697 CF8G3E 24971332 IC50 = 365000 nM T89697 CPR02N 24971333 IC50 = 734000 nM T89697 C10SAI 24971370 IC50 = 4950 nM T89697 CV6L8H 25141140 Ki = 76300 nM T89697 C1XU4T 25141142 Ki = 87100 nM T89697 CQJ8F1 25211983 IC50 = 127 nM T89697 C0ZJY1 25211984 IC50 = 188 nM T89697 CO2GF9 25241857 IC50 = 5400 nM T89697 C0DT1U 25241896 IC50 = 2200 nM T89697 CPC12H 25241897 IC50 = 900 nM T89697 C9OWU5 26921488 IC50 > 30000 nM T89697 CX8T3C 28934713 IC50 > 50000 nM T89697 CUGD12 28934715 IC50 = 34000 nM T89697 CJ9S5L 28934757 IC50 > 50000 nM T89697 CJU84V 28934769 IC50 > 50000 nM T89697 CZ98CD 28934783 IC50 = 1200 nM T89697 CF8CJ7 30762236 IC50 > 30000 nM T89697 CH0DU1 35353466 IC50 = 99350 nM T89697 C8JMZ6 35354409 IC50 = 99830 nM T89697 CE8F0K 36688758 IC50 = 54100 nM T89697 CN19VO 40418972 IC50 = 3800 nM T89697 C4S7PI 43348154 IC50 = 34000 nM T89697 CL04IU 44156271 IC50 = 14000 nM T89697 CPN0X1 44251142 Ki = 11550 nM T89697 C4G3PD 44406794 Ki = 28380 nM T89697 CX5Y4V 44406795 Ki = 20480 nM T89697 C7Q8JF 44406806 Ki = 36950 nM T89697 CR57ND 44406812 Ki = 363600 nM T89697 CVH98E 44457253 IC50 = 82 nM T89697 CVRQ27 44457255 IC50 = 186 nM T89697 CS17JV 44457280 IC50 = 55 nM T89697 C24PTC 44457418 IC50 = 1500 nM T89697 CS7I1E 44457419 IC50 = 512 nM T89697 CT0YX5 44457436 IC50 = 2120 nM T89697 CT8K3L 44457437 IC50 = 1090 nM T89697 CI2VN4 44457447 IC50 = 3960 nM T89697 C87CKB 44457448 IC50 = 360 nM T89697 C7W8KH 44465701 IC50 = 450 nM T89697 CO15EU 44465944 IC50 > 1000000 nM T89697 C97EPW 44465950 IC50 = 400000 nM T89697 C1SF4O 44465951 IC50 = 90000 nM T89697 C04XGN 44465952 IC50 = 60000 nM T89697 C0JPM6 44466194 IC50 = 105000 nM T89697 C3BVF5 44466197 IC50 = 5000 nM T89697 CT1KO3 44466198 IC50 = 200000 nM T89697 C15FTG 44467660 IC50 = 9100 nM T89697 CEQ9F7 44467799 IC50 = 18000 nM T89697 C8C4GX 44468002 IC50 = 23000 nM T89697 CA60ES 44597169 IC50 > 20000 nM T89697 CWC4K1 44597274 IC50 = 1400 nM T89697 CM7T5C 44597275 IC50 = 1400 nM T89697 C2QT3S 44597276 IC50 > 2000 nM T89697 CF8DA5 44597277 IC50 > 2000 nM T89697 C2AP6Q 44819148 IC50 = 22400 nM T89697 CA0KJ8 44819149 IC50 = 12600 nM T89697 CZ3M0U 45158558 IC50 = 570 nM T89697 CW9B1I 45248340 IC50 = 18600 nM T89697 CPLJ59 45482936 IC50 = 11900 nM T89697 C4GO2W 45482946 IC50 = 4200 nM T89697 C24MGQ 45482949 IC50 = 7100 nM T89697 CU3F6W 45487175 IC50 = 50000 nM T89697 CL93SV 45487181 IC50 = 200 nM T89697 C6U2HB 45487187 IC50 = 50000 nM T89697 C7O5EN 45487189 IC50 = 44000 nM T89697 C2ASP5 45487202 IC50 = 40000 nM T89697 CYD0A1 45487207 IC50 = 50000 nM T89697 C2D3ZL 45487229 IC50 = 25000 nM T89697 CLWY27 46180669 IC50 = 520 nM T89697 C6HTU7 46834223 IC50 = 1371000 nM T89697 CQL2S9 46913822 IC50 = 24600 nM T89697 C96QOX 47827438 IC50 = 90 nM T89697 C7T2OH 47827446 IC50 = 961 nM T89697 C9BM5X 49866156 IC50 > 20000 nM T89697 CWOF35 49866158 IC50 > 20000 nM T89697 C2NJ3B 51003508 IC50 = 14000 nM T89697 CMF2O6 52912227 IC50 < 1000 nM T89697 CQP52L 52918052 IC50 = 36000 nM T89697 C06VWA 52932742 IC50 < 1000 nM T89697 C58PSL 52935731 IC50 = 1700 nM T89697 C7P1KN 52936167 IC50 = 1700 nM T89697 CEQN27 52936621 Ki > 1000 nM T89697 CZ0CG8 52942238 IC50 = 880 nM T89697 CFR5M9 53316976 IC50 = 37000 nM T89697 CO2KF5 53317021 IC50 = 96000 nM T89697 CW6Q5U 53317048 IC50 = 37000 nM T89697 CD1J7C 53318255 IC50 = 45000 nM T89697 CKF1H7 53318256 IC50 = 141000 nM T89697 CFB26Q 53318297 IC50 = 83000 nM T89697 C2ZLA8 53318331 IC50 = 43000 nM T89697 CW9T8K 53319620 IC50 = 34000 nM T89697 CS3Y6N 53319657 IC50 = 18000 nM T89697 CS5T9R 53319675 IC50 = 82000 nM T89697 CF6EU4 53320957 IC50 = 87000 nM T89697 CD0IC5 53322284 IC50 = 153000 nM T89697 CSO21L 53323252 IC50 = 29000 nM T89697 CG1R0E 53323675 IC50 = 13100 nM T89697 C7RKN6 53324267 IC50 = 26200 nM T89697 C7BA9R 53324928 IC50 = 58000 nM T89697 CP2AK1 53324929 IC50 = 49000 nM T89697 CK4LN0 53324956 IC50 = 63000 nM T89697 CAB8U0 53326252 IC50 = 139000 nM T89697 CQ4PM6 55254080 IC50 = 490 nM T89697 CT5M9H 56659238 Ki = 40000 nM T89697 CKG5F8 56666431 IC50 = 92000 nM T89697 CP6V9F 57408307 IC50 = 21000 nM T89697 CA19IT 57611775 EC50 = 1260 nM T89697 CA3XG9 58294074 IC50 = 6600 nM T89697 CR57BA 58294080 EC50 = 2400 nM T89697 CGQ3X8 58294086 EC50 = 110000 nM T89697 CPAV97 58294088 IC50 = 3800 nM T89697 C8EYR1 58294092 IC50 > 1000000 nM T89697 C26VNU 58294099 IC50 = 187000 nM T89697 C4LD1V 58294110 IC50 = 312000 nM T89697 COXA92 58294117 IC50 = 300 nM T89697 CZXO68 58294132 IC50 = 5100 nM T89697 CJL85W 58294141 IC50 = 7200 nM T89697 C01SLN 58294147 IC50 = 960 nM T89697 CRL75F 58294169 IC50 = 7800 nM T89697 CU0V3W 58294216 EC50 = 1700 nM T89697 C63ZDL 58294226 IC50 = 44000 nM T89697 CLI6P9 58294227 IC50 > 1000000 nM T89697 CO05DE 58693509 IC50 = 1000 nM T89697 CVJ0N6 60154724 IC50 = 4300 nM T89697 CA1TW8 60154725 IC50 = 6400 nM T89697 CA8W4D 60154726 IC50 = 23000 nM T89697 C6AMR4 60154727 IC50 = 72000 nM T89697 C0ZP8T 60154728 IC50 = 1200000 nM T89697 CU12TW 60154729 IC50 = 3000000 nM T89697 CRKM01 60154730 IC50 = 3200000 nM T89697 CW0FS2 60156091 IC50 = 1100 nM T89697 CDM64W 60156092 IC50 = 2800 nM T89697 CS31CB 60156093 IC50 = 3300 nM T89697 C2LSA3 60156094 IC50 = 7400 nM T89697 CA34YM 60156095 IC50 = 56000 nM T89697 CP34LY 60156096 IC50 = 1800000 nM T89697 CK9JV7 60623327 IC50 = 53130 nM T89697 CQ0G4K 60623350 IC50 = 49250 nM T89697 CSVT86 66553577 IC50 = 10000 nM T89697 CP59KG 66553578 IC50 = 11000 nM T89697 CD2H5Z 66553579 IC50 = 53000 nM T89697 C3C2VH 66553580 IC50 = 29000 nM T89697 C1LB6D 66558197 IC50 = 610 nM T89697 CHX38T 66558199 EC50 = 5900 nM T89697 CU4E2L 66558294 IC50 = 1100 nM T89697 CN91RJ 66558377 EC50 = 5400 nM T89697 C7UKS4 66558379 EC50 = 1100 nM T89697 C9ML2G 66558380 EC50 = 15000 nM T89697 CA4B9P 66558554 IC50 = 1000 nM T89697 CCK6E5 66558639 IC50 = 45 nM T89697 C35NBR 66558640 IC50 = 2400 nM T89697 CK2ZH4 66558723 IC50 = 2900 nM T89697 C8PJ5X 66558811 IC50 = 370 nM T89697 CZ1R2N 66558888 IC50 = 8800 nM T89697 CFM1C3 66760716 IC50 = 3400 nM T89697 C9XC3P 66761410 IC50 = 1400 nM T89697 CBZT64 66761654 IC50 = 2700 nM T89697 CQO09P 67036471 IC50 = 53000 nM T89697 CBH06U 67131986 IC50 = 340 nM T89697 CL0ZD8 67132094 IC50 = 2400 nM T89697 CIC2O5 67132131 IC50 = 1600 nM T89697 C9XRU4 67132184 IC50 = 900 nM T89697 CJ6YI2 67207384 IC50 = 47000 nM T89697 C69FWP 67222089 IC50 > 1000000 nM T89697 C27GIY 68348080 EC50 = 7900 nM T89697 C46KPQ 68348135 IC50 = 32000 nM T89697 CC42EQ 68348137 IC50 = 154000 nM T89697 CX4Y2I 69476274 IC50 = 15000 nM T89697 CA92SK 70874201 IC50 = 3400 nM T89697 CUCQ24 70874317 EC50 = 93 nM T89697 CSO9W5 70874322 EC50 = 490 nM T89697 C1IJ0W 70874391 EC50 = 780 nM T89697 CO3Y9B 70874393 EC50 = 510 nM T89697 C8LCK6 70874412 EC50 = 2200 nM T89697 C1H7VK 70874453 IC50 = 19 nM T89697 CJF91M 70874544 IC50 = 46 nM T89697 C9EWB8 70874603 EC50 = 200 nM T89697 C8CMD0 70874604 IC50 < 1000 nM T89697 C82PUD 70874605 EC50 = 78 nM T89697 CMW8S2 70874703 EC50 = 2700 nM T89697 CIW3M7 70874768 EC50 = 725 nM T89697 CQC35B 70874783 IC50 = 110 nM T89697 C8Q4LJ 70874786 EC50 = 130 nM T89697 CKQ5U7 70874818 IC50 = 1000 nM T89697 CA45OH 70874831 EC50 = 240 nM T89697 C83RQG 70874868 EC50 = 820 nM T89697 CCW4B5 70874889 EC50 = 6700 nM T89697 C2TZ8D 70874895 EC50 = 760 nM T89697 CF1G3K 70874916 IC50 = 200 nM T89697 CPLT90 70874941 EC50 = 230 nM T89697 CJ24YM 70914178 IC50 = 468 nM T89697 CJ80SV 70914181 IC50 = 127000 nM T89697 C30AJI 70914208 IC50 = 50 nM T89697 C7BDH0 70914212 IC50 = 1500 nM T89697 C71AZM 70914219 EC50 = 1300 nM T89697 C2TC8W 70914230 Ki = 5.8 nM T89697 C8V5NF 70914234 EC50 = 220 nM T89697 CP8HI7 70914358 IC50 = 700 nM T89697 CJN0M5 70925897 EC50 = 6100 nM T89697 CNUF17 71458329 IC50 = 47000 nM T89697 CN8Q3X 74221589 IC50 < 100 nM T89697 CTL8X2 75202661 IC50 = 100 nM T89697 C5YFU8 75202920 IC50 = 1000 nM T89697 C6HPF7 75202926 IC50 = 1000 nM T89697 C2D6KV 75203053 IC50 < 100 nM T89697 CVLP16 75203175 IC50 = 100 nM T89697 CQ5LH4 75405939 IC50 = 64 nM T89697 C56YXL 76320783 IC50 = 24.3 nM T89697 C40EJG 76324723 IC50 = 6000 nM T89697 CRT2C5 76327994 IC50 = 451000 nM T89697 C1HXJ9 76327995 IC50 = 185 nM T89697 CFT9L1 76334268 IC50 = 1600 nM T89697 C2JYL9 77050772 IC50 = 240 nM T89697 CF9X8G 77050773 IC50 = 240 nM T89697 CXC63V 77952883 EC50 = 1100 nM T89697 CZL45X 78425875 IC50 = 0.5 nM T89697 CT7VC8 84374905 IC50 = 3109.3 nM T89697 CGT4O9 85469240 IC50 = 1870 nM T89697 C8T0MJ 85469241 IC50 = 1800 nM T89697 C5SWD9 85469242 IC50 = 590 nM T89697 CA5CG1 85469243 IC50 = 760 nM T89697 C5R6WS 85469292 IC50 = 2960 nM T89697 CWN56M 85626388 IC50 = 4730 nM T89697 C8T0CH 86240712 IC50 > 50000 nM T89697 C1Z2TQ 86240717 IC50 = 1800 nM T89697 CO82UY 86240725 IC50 = 2100 nM T89697 CSGQ82 86240731 IC50 = 54000 nM T89697 CT8SW0 86764097 IC50 = 2400 nM T89697 C1WBQ3 86764098 IC50 = 70 nM T89697 CRL9C7 86764205 IC50 = 120 nM T89697 CI05RT 89052784 IC50 = 20370 nM T89697 CH8JT1 89052953 IC50 = 120000 nM T89697 C7VB9Z 89999091 EC50 = 220 nM T89697 CC32EF 90423425 IC50 < 200 nM T89697 C39EMN 90644514 IC50 > 50000 nM T89697 CPV54D 90644515 IC50 > 50000 nM T89697 C0FH2K 90644516 IC50 > 50000 nM T89697 C7Z5NK 90718185 IC50 = 4 nM T89697 C3Z8YX 91758737 IC50 = 20 nM T89697 C3BXV4 101894468 IC50 = 110 nM T89697 CBF1P2 101894469 IC50 = 4000 nM T89697 CJ19AQ 102128193 Ki = 35 nM T89697 C6AFB0 102128195 Ki = 35 nM T89697 C9VZ4F 117620853 EC50 > 10000 nM T89697 C46AOF 117704863 IC50 < 200 nM T89697 CI0Y8F 117779240 IC50 = 350 nM T89697 CJH1Z4 117800109 IC50 = 5 nM T89697 CP75IE 117927565 IC50 = 661 nM T89697 C7L6SF 117927575 IC50 = 76 nM T89697 CQZI27 117927580 IC50 = 13 nM T89697 C4YE0X 118511968 IC50 = 13000 nM T89697 CUAP64 118511969 IC50 > 50000 nM T89697 CS74VJ 118511985 IC50 = 620 nM T89697 CDP71A 118511986 IC50 = 290 nM T89697 C37OSM 118511993 IC50 > 50000 nM T89697 CKG90Q 118512005 IC50 > 50000 nM T89697 C4SWU1 118512015 IC50 = 1200 nM T89697 CN98IG 118512017 IC50 = 120 nM T89697 C50AFG 118512030 IC50 = 1700 nM T89697 C0MEC2 118512032 IC50 = 46000 nM T89697 C4J7UP 118512042 IC50 = 580 nM T89697 C41XHC 118512043 IC50 = 490 nM T89697 C4Z8QL 118512052 IC50 = 8000 nM T89697 CJ6B7A 118512054 IC50 = 2200 nM T89697 CM1DS2 118512060 IC50 > 50000 nM T89697 CPT8K5 118512063 IC50 = 4600 nM T89697 CPFQ23 118512079 IC50 = 3400 nM T89697 CEK8O4 118512091 IC50 = 1700 nM T89697 C8IUD4 118569598 IC50 < 1000 nM T89697 CMRV56 118706416 IC50 = 80 nM T89697 CK9GQ7 118706833 IC50 = 43 nM T89697 CG1A3O 118706834 IC50 = 59 nM T89697 C32BDE 118706835 EC50 = 296 nM T89697 C4Z8XI 118706836 EC50 = 1171 nM T89697 C0IHA8 118706837 IC50 = 254 nM T89697 C2T8ZF 118706838 EC50 = 1393 nM T89697 CHE7P0 118706839 EC50 = 181 nM T89697 CFU73S 118706840 EC50 = 142 nM T89697 CD5YM8 118706841 EC50 = 85 nM T89697 C9KME7 118706842 IC50 = 122 nM T89697 C5O2BI 118706843 IC50 = 255 nM T89697 CT6L3M 118706844 EC50 = 2494 nM T89697 CNMZ08 118706845 EC50 = 2588 nM T89697 C2FN6H 118706846 EC50 = 187 nM T89697 COU9T3 118706847 EC50 = 130 nM T89697 CU40NV 118706848 EC50 = 84 nM T89697 CG9B5A 118706849 EC50 = 2229 nM T89697 C5Q3DP 118706850 IC50 = 608 nM T89697 C2GLY9 118706851 IC50 = 247 nM T89697 C9G8WM 118706944 EC50 = 508 nM T89697 CHQV01 118706945 EC50 = 374 nM T89697 CW2HM0 118706946 EC50 = 134 nM T89697 CTB7D6 118706947 EC50 = 465 nM T89697 COZV69 118706948 EC50 = 187 nM T89697 CTF8K6 118706949 EC50 = 183 nM T89697 CK5W7Z 118706950 IC50 = 125 nM T89697 CT87ZE 118706951 EC50 = 172 nM T89697 C1REB5 118706952 IC50 = 4055 nM T89697 C26LNH 118708818 IC50 = 84000 nM T89697 CV8M5E 118716422 IC50 = 18000 nM T89697 CD08UQ 118716423 IC50 > 100000 nM T89697 C0NHP3 118716424 IC50 > 100000 nM T89697 C0LN8P 118716425 IC50 > 100000 nM T89697 CYI8E6 118716426 IC50 > 100000 nM T89697 CMX5F2 118716427 IC50 = 24000 nM T89697 CT9HZ8 118716428 IC50 = 56000 nM T89697 CIOK68 118716429 IC50 = 8100 nM T89697 C1OMC9 118716430 IC50 = 5500 nM T89697 C0TA6G 118716431 IC50 > 100000 nM T89697 CHOC51 118716432 IC50 = 3500 nM T89697 CA6NH1 118716433 IC50 = 1900 nM T89697 C0M2FU 118716434 IC50 = 3600 nM T89697 CV7DW6 118716435 IC50 = 220 nM T89697 C41QXJ 118716436 IC50 = 750 nM T89697 CF16UH 118716437 IC50 = 1800 nM T89697 CDK5J0 118716438 IC50 = 120 nM T89697 CW3HZ6 118716439 IC50 = 160 nM T89697 C6AI5J 118716440 IC50 = 190 nM T89697 C8YUR0 118716441 IC50 = 77 nM T89697 CI0CN3 118720652 IC50 = 1300 nM T89697 CRH1D8 121332565 IC50 > 1000 nM T89697 C3BMW5 121332569 IC50 = 50 nM T89697 CK82EH 121332589 IC50 = 830 nM T89697 CU6JL0 121332595 IC50 = 690 nM T89697 C65ZYO 121332604 IC50 = 22 nM T89697 CK4W2N 121332617 IC50 = 250 nM T89697 C6CTF1 121332626 IC50 = 540 nM T89697 C5YS9V 121332627 IC50 = 160 nM T89697 CZ2TG3 121332650 IC50 = 1800 nM T89697 CNMK19 121332652 IC50 = 330 nM T89697 C92NOH 121332654 IC50 = 100 nM T89697 CF2Y4A 121332661 IC50 = 790 nM T89697 C5CH7A 121332672 IC50 = 2900 nM T89697 C2Z9YC 121332674 IC50 = 280 nM T89697 CF1C2J 121332677 IC50 = 340 nM T89697 CDL5N6 121332679 IC50 = 1000 nM T89697 C0O2WL 121332691 IC50 = 62 nM T89697 CN0UL6 121332697 IC50 = 2100 nM T89697 CB5LH6 121332700 IC50 = 570 nM T89697 C96RZJ 121332707 IC50 = 1800 nM T89697 CRG82W 121332712 IC50 = 840 nM T89697 CLD6W9 121332721 IC50 = 2600 nM T89697 CNBH32 121332727 IC50 = 49 nM T89697 C0M1TY 121332731 IC50 = 1500 nM T89697 C2EQP8 121332773 IC50 = 50 nM T89697 CMP01Q 121354659 IC50 = 5 nM T89697 C8GXR1 121469000 IC50 = 42 nM T89697 CFQ9P6 121469056 IC50 = 159 nM T89697 C7J0RI 121469136 IC50 = 348 nM T89697 C7OQU1 121469151 IC50 = 14 nM T89697 CW7N8S 121469162 IC50 = 504 nM T89697 CND02B 121469183 IC50 = 45 nM T89697 CJ85LD 121469184 IC50 = 23 nM T89697 C9Q0TD 121469223 IC50 > 1000 nM T89697 CX3Q8C 121469247 IC50 = 600 nM T89697 CS6PA4 121469296 IC50 > 1000 nM T89697 CUP95H 121474590 IC50 > 1000 nM T89697 CSF24O 122193552 IC50 = 3163 nM T89697 C25XGV 122193553 IC50 > 10000 nM T89697 CV30GB 122193590 IC50 = 1242 nM T89697 C4RSB3 122193591 IC50 = 2323 nM T89697 C4N9HG 122193592 IC50 = 977 nM T89697 C8A0DL 122193593 IC50 = 1928 nM T89697 CR27QH 122193594 IC50 = 602 nM T89697 CXY02W 122193595 IC50 = 936 nM T89697 CJ6RO8 122193596 IC50 = 640 nM T89697 CL7S4T 122193597 IC50 = 1097 nM T89697 CCL63T 122193598 IC50 = 982 nM T89697 CP93QC 122193599 IC50 = 2069 nM T89697 CIDM29 122193600 IC50 = 1593 nM T89697 C2U6VA 122193601 IC50 = 921.8 nM T89697 CPG6T0 122368191 IC50 = 48 nM T89697 CC6VJ5 122525709 IC50 = 180 nM T89697 CY0X9D 122525711 IC50 = 20 nM T89697 CZE79W 122525712 IC50 = 680 nM T89697 C51WNS 122606362 IC50 = 20 nM T89697 CGO29F 122608329 IC50 = 130 nM T89697 CXS30F 122650362 IC50 > 10000 nM T89697 CF9Q1R 122650368 IC50 > 10000 nM T89697 CU2K4P 122650372 IC50 = 26 nM T89697 C3RCU4 122650378 IC50 = 21 nM T89697 C3LY8T 122650476 IC50 = 81 nM T89697 CP9EY1 122650500 IC50 = 167 nM T89697 CN6MK9 122650505 IC50 = 87 nM T89697 CHZY51 122650508 IC50 = 79 nM T89697 CS47AD 122650581 IC50 = 8 nM T89697 C3YM4T 124927661 IC50 = 289.5 nM T89697 CWN4D0 125315466 IC50 = 217000 nM T89697 CGP91U 127026194 IC50 = 77 nM T89697 C1XVD6 127026502 IC50 = 68.1 nM T89697 C86NVH 127026503 EC50 = 231.4 nM T89697 CJL27E 127027129 EC50 = 30.6 nM T89697 CY7SM8 127027130 EC50 = 36.4 nM T89697 CDV03C 127027131 EC50 = 67 nM T89697 C36HFU 127027132 EC50 = 211.5 nM T89697 C9A4RT 127027138 EC50 = 63.1 nM T89697 CY6M9H 127027139 EC50 = 68.4 nM T89697 C8YKZ6 127027140 EC50 = 134.9 nM T89697 CEU96I 127027427 IC50 = 111.8 nM T89697 CG08KV 127028367 IC50 = 10000 nM T89697 CW7A2Q 127028368 IC50 = 10000 nM T89697 C51QDO 127028910 IC50 > 10000 nM T89697 C9QVB4 127036449 EC50 > 10000 nM T89697 CK6SC5 127036625 IC50 = 48000 nM T89697 C1HUY5 127036630 IC50 > 10000 nM T89697 C23XQU 127036787 IC50 = 1139 nM T89697 CQ8U6F 127037839 IC50 = 1100 nM T89697 C7ZC9Q 127037878 EC50 = 67.6 nM T89697 CIA42L 127038189 IC50 = 20000 nM T89697 CIQ15P 127038190 IC50 = 730 nM T89697 C46ISV 127038222 IC50 = 82 nM T89697 CV7FO1 127038232 IC50 = 4600 nM T89697 CX0JH6 127038891 IC50 = 5200 nM T89697 C3YQJ0 127039199 IC50 = 4200 nM T89697 C2S6BH 127039223 IC50 = 1700 nM T89697 C9RB4I 127039229 IC50 = 19000 nM T89697 C9MK6V 127039238 IC50 = 61000 nM T89697 C79HKG 127039239 IC50 = 490 nM T89697 CSG51N 127039240 IC50 = 570 nM T89697 C7T0HM 127039543 IC50 = 55000 nM T89697 CGL2K6 127039550 IC50 = 26000 nM T89697 CV5I4T 127039862 IC50 = 75.8 nM T89697 CS1X3N 127040995 IC50 = 7700 nM T89697 CT4RU6 127041800 IC50 > 10000 nM T89697 CB2S4P 127042503 IC50 < 1000 nM T89697 C3SXY7 127046261 IC50 > 30000 nM T89697 CM4R5A 127046282 IC50 > 30000 nM T89697 C75UNV 127046283 IC50 > 30000 nM T89697 CAHF82 127046284 IC50 > 30000 nM T89697 C6XZ7M 127046780 IC50 > 30000 nM T89697 C6J3PV 127046921 IC50 > 30000 nM T89697 C57UIH 127047228 IC50 = 3500 nM T89697 CDKF67 127047240 IC50 > 30000 nM T89697 CZ4SV2 127047241 IC50 = 3400 nM T89697 C2JTQ3 127047242 IC50 > 30000 nM T89697 C5P4JH 127047325 IC50 = 1500 nM T89697 CHZA26 127047364 IC50 > 30000 nM T89697 CGE49W 127047365 IC50 > 30000 nM T89697 CIX95S 127047490 IC50 > 30000 nM T89697 CE94JR 127047748 IC50 = 6300 nM T89697 CV1X0F 127047886 IC50 = 1700 nM T89697 CM2NL5 127048012 IC50 = 4700 nM T89697 CI38DX 127048013 IC50 = 4900 nM T89697 C7XW2S 127048014 IC50 > 30000 nM T89697 C9L7ZW 127048015 IC50 > 30000 nM T89697 C7F3TB 127048016 IC50 = 2800 nM T89697 C6JZ9N 127048017 IC50 = 3800 nM T89697 CK5C8N 127048018 IC50 = 5400 nM T89697 CJ43QC 127048019 IC50 = 7200 nM T89697 C60WCP 127048119 IC50 = 2100 nM T89697 CY7G4D 129282405 EC50 = 720 nM T89697 CQ97RT 129282436 EC50 = 1400 nM T89697 CL9J8N 129282617 EC50 = 2200 nM T89697 CP09TF 129282671 EC50 = 2900 nM T89697 C42ZDX 129282689 EC50 = 1600 nM T89697 C3GA7K 129282703 EC50 = 4500 nM T89697 CV28YE 129282706 EC50 = 1300 nM T89697 C7LG2X 129282851 EC50 = 20000 nM T89697 C3SGN0 129282870 EC50 = 1400 nM T89697 CU70NI 129282903 EC50 > 25000 nM T89697 C3CH6E 129283030 EC50 = 13000 nM T89697 C7FXS8 129283166 EC50 = 880 nM T89697 C32WDC 129283174 EC50 = 240 nM T89697 C9HZ2S 129283211 EC50 = 4600 nM T89697 C5L7MR 129283737 EC50 = 970 nM T89697 CE19JM 129296385 EC50 = 800 nM T89697 C56BAE 129296459 EC50 > 25000 nM T89697 COU73Q 132528948 IC50 = 5300 nM T89697 CDMH46 132606955 IC50 = 560 nM T89697 CNX3D4 134130983 Ki = 35 nM T89697 CCX46W 134131669 Ki = 35 nM T89697 C0KX5B 134132343 Ki = 35 nM T89697 C95RJQ 134132658 Ki = 35 nM T89697 CC47DZ 134132888 Ki = 35 nM T89697 CCS0M6 134133190 Ki = 35 nM T89697 C5UM0A 134135015 Ki = 35 nM T89697 CPR5A4 134136354 Ki = 35 nM T89697 C46MUG 134136717 Ki = 35 nM T89697 CQZB67 134137635 Ki = 35 nM T89697 C8QOD7 134138847 Ki = 35 nM T89697 CNE10R 134139474 Ki = 35 nM T89697 CVB51Y 134141021 Ki = 35 nM T89697 C2QL6D 134142610 Ki = 35 nM T89697 CQD8V6 134142830 Ki = 35 nM T89697 C0HKW5 134143335 Ki = 35 nM T89697 CV5XQ0 134143523 Ki = 35 nM T89697 C4KDS5 134145910 Ki = 35 nM T89697 C2HJ8Z 134146158 Ki = 35 nM T89697 C8D9KR 134146460 Ki = 35 nM T89697 CZ73SH 134147587 Ki = 35 nM T89697 CSUE71 134149657 Ki = 35 nM T89697 CH3C9P 134150058 Ki = 35 nM T89697 CI69YJ 134150572 Ki = 35 nM T89697 CB87LJ 134152033 Ki = 35 nM T89697 CS8W4E 134153755 Ki = 35 nM T89697 CM62BZ 134154095 Ki = 35 nM T89697 C15WLQ 134154247 Ki = 35 nM T89697 C9WQ6T 134155013 Ki = 35 nM T89697 CH7CX3 134155058 Ki = 35 nM T89697 CIV1X4 134156014 Ki = 35 nM T89697 CCP20Z 134156288 Ki = 35 nM T89697 CA6C5U 134157947 Ki = 35 nM T89697 C9ZEJ4 134462563 IC50 = 568 nM T89697 CO1YD8 135401349 IC50 > 30000 nM T89697 CCJ85U 135412567 IC50 = 1240 nM T89697 CPK9A8 135420064 IC50 = 8600 nM T89697 CFWY62 135424939 IC50 = 1500 nM T89697 CG81PH 135424940 IC50 = 270 nM T89697 CDC15J 135424941 IC50 = 19 nM T89697 CUK07Z 135424945 IC50 = 6800 nM T89697 C3P7VU 135424946 IC50 = 970 nM T89697 CB9Q2N 135424953 IC50 = 14 nM T89697 CY20NS 135424981 IC50 = 14 nM T89697 CIT4U8 135437626 IC50 > 30000 nM T89697 CVQ6I5 135442567 IC50 = 2850 nM T89697 C9L3NY 135465938 IC50 = 21100 nM T89697 CHI9L5 135472487 IC50 > 30000 nM T89697 CWV63H 135478380 IC50 = 10300 nM T89697 CXE5S3 135482065 IC50 = 1700 nM T89697 CRYK71 135491081 IC50 = 11300 nM T89697 C0A5WI 135510775 IC50 = 73 nM T89697 CNY13I 135510784 IC50 = 54 nM T89697 CEU6N4 135533698 IC50 > 30000 nM T89697 CW5LN1 135533790 IC50 = 2100 nM T89697 CKT9M6 135567420 IC50 = 2.8 nM T89697 CI2GV6 135588554 IC50 > 30000 nM T89697 CZJ24D 135588681 IC50 = 4800 nM T89697 CXD4W7 135611181 IC50 = 6000 nM T89697 CS0DA5 135741412 IC50 = 10 nM T89697 CASN86 135743630 IC50 > 100000 nM T89697 CK7RW0 135821912 IC50 > 30000 nM T89697 CF95ES 135895369 IC50 = 100 nM T89697 CO56EF 135895372 IC50 = 120 nM T89697 CA2M7V 135899518 Ki = 367000 nM T89697 C7H3IM 135905429 IC50 = 100 nM T89697 C7Y0PK 135936842 IC50 = 2100 nM T89697 C9KHP8 135981331 IC50 = 53 nM T89697 CDH36U 136036203 Ki = 197000 nM T89697 C2L6CP 136099973 IC50 = 280 nM T89697 CU13NF 136123535 IC50 = 7000 nM T89697 C98DMB 136898218 IC50 = 98 nM T89697 C9V1YI 137223162 IC50 = 12 nM T89697 CW2RC3 137245067 IC50 = 35 nM T89697 CNGL30 137250365 IC50 = 17.9 nM T89697 C7EJZ4 137297236 IC50 = 16 nM T89697 CO32JA 137297260 IC50 = 52 nM T89697 C15UNK 137297264 IC50 = 373 nM T89697 CU34ZO 137297270 IC50 = 23070 nM T89697 C8VQ9X 137297286 IC50 > 10000 nM T89697 CVDH54 137297313 IC50 = 2748 nM T89697 CX7L0Y 137297324 IC50 = 2094 nM T89697 CWCD40 137297341 IC50 = 26 nM T89697 C1ARX6 137297350 IC50 = 26 nM T89697 C31AZO 137297358 IC50 = 20 nM T89697 C4SM2V 137297442 IC50 = 853 nM T89697 CZ7MF4 137297447 IC50 = 18 nM T89697 CQM4I6 137297497 IC50 = 1235 nM T89697 CL5Q1S 137386090 IC50 = 151.5 nM T89697 C5LPK1 137386135 IC50 = 55.7 nM T89697 CX8ZD9 137386139 IC50 = 14.4 nM T89697 CY73OP 137386143 IC50 = 17.1 nM T89697 CO5SY2 137386223 IC50 = 18.8 nM T89697 CKHW29 137386229 IC50 = 35.6 nM T89697 C2A3WV 137386236 IC50 = 251 nM T89697 CJ73IG 137390209 EC50 = 420 nM T89697 CA5OY1 137628667 EC50 = 410 nM T89697 C4HJU2 137631563 IC50 = 23000 nM T89697 CB3RA0 137632598 IC50 = 366000 nM T89697 CK5TL4 137634430 EC50 = 15310 nM T89697 CMU1O6 137634654 IC50 > 5000 nM T89697 CK8A9L 137637814 IC50 = 5255 nM T89697 C85QBH 137639169 IC50 = 47000 nM T89697 C4JM6K 137639484 IC50 = 9784 nM T89697 C2B3NF 137640065 IC50 = 22 nM T89697 CXJH24 137640336 IC50 = 6000 nM T89697 C8RVQ3 137641068 IC50 = 9700 nM T89697 CGL56P 137643600 IC50 = 41000 nM T89697 CY6R3Q 137647941 IC50 = 210 nM T89697 CQ5G4T 137650989 IC50 = 100 nM T89697 C0K9MI 137651594 EC50 = 17540 nM T89697 CFQ2V0 137655049 IC50 = 4500 nM T89697 CI8A1Y 137655874 IC50 = 2400 nM T89697 C46BDF 137657792 IC50 = 172000 nM T89697 COED37 137661429 IC50 = 27600 nM T89697 C96QPV 137662004 IC50 = 87 nM T89697 CQ89OP 138737778 IC50 = 230 nM T89697 CZHY27 138737927 IC50 = 15 nM T89697 C1WFB4 138737941 IC50 = 9.3 nM T89697 C39POY 139507046 IC50 = 14 nM T89697 CD29IP 139507088 IC50 = 21 nM T89697 CEFG75 141483091 IC50 = 14560 nM T89697 C5L2QN 141483093 IC50 = 99940 nM T89697 C3GQC2 141483094 IC50 = 31820 nM T89697 CKY6N8 141483096 IC50 = 6400 nM T89697 CRT49I 141483097 IC50 = 80780 nM T89697 C7LPO8 141483098 IC50 > 100000 nM T89697 CB0GA4 141483099 IC50 = 28490 nM T89697 CHA20C 141483100 IC50 > 100000 nM T89697 CH60KW 141501915 IC50 = 50900 nM T89697 CV91LK 141501916 IC50 = 74390 nM T89697 CBE81C 141501917 IC50 = 39040 nM T89697 CCJV28 141501918 IC50 = 14980 nM T89697 C69RFM 141501919 IC50 = 64470 nM T89697 C81KPZ 141501920 IC50 = 22720 nM T89697 CCN50V 141501921 IC50 = 25930 nM T89697 CA1YE4 141501922 IC50 = 95070 nM T89697 CS9OX0 141501923 IC50 = 53930 nM T89697 C5HW7N 141501924 IC50 = 69440 nM T89697 CNL6A2 141501925 IC50 = 840 nM T89697 CF41KS 141501926 IC50 = 33100 nM T89697 C8BVO4 141501927 IC50 = 21930 nM T89697 CI90SH 141501931 IC50 = 77540 nM T89697 CZ6E1A 141501932 IC50 = 60560 nM T89697 CX7K2H 141514151 IC50 = 260.3 nM T89697 C7XGA5 141744794 IC50 > 10000 nM T89697 C5W6QL 141744795 IC50 = 250 nM T89697 CS0VF4 141744796 IC50 = 6780 nM T89697 CEF7Q9 141744797 IC50 > 10000 nM T89697 CS1N8K 141744798 IC50 > 10000 nM T89697 CRK06D 141744799 IC50 = 4840 nM T89697 C78ELY 141744800 IC50 = 9600 nM T89697 C03BNS 141744801 IC50 = 78 nM T89697 CDV98B 141744802 IC50 = 160 nM T89697 CY1CJ9 141744803 IC50 > 10000 nM T89697 CX37LU 141744804 IC50 > 10000 nM T89697 C3A8DH 141744805 IC50 > 10000 nM T89697 CDAP21 141744806 IC50 = 6110 nM T89697 C8VTK2 141744807 IC50 = 630 nM T89697 CJB0H5 141744808 IC50 = 240 nM T89697 C4LW7Q 141744809 IC50 = 2090 nM T89697 C7LA5F 141744810 IC50 = 8190 nM T89697 CLUM57 141744811 IC50 > 10000 nM T89697 CAM31S 141744813 IC50 > 10000 nM T89697 CMKN19 141744814 IC50 > 10000 nM T89697 CU2Q6E 141744815 IC50 > 10000 nM T89697 C9YT2N 141744816 IC50 > 10000 nM T89697 C9KVZ4 141744817 IC50 = 74 nM T89697 C78GZL 141744818 IC50 = 97 nM T89697 C7JYI3 141744820 IC50 = 82 nM T89697 C0EDU6 141744821 IC50 = 8270 nM T89697 CGO28U 141744823 IC50 = 3210 nM T89697 CE5O2V 141744824 IC50 > 10000 nM T89697 CB8X5H 141744825 IC50 = 1510 nM T89697 C7Q2WE 141744826 IC50 = 3540 nM T89697 C37XEL 141744827 IC50 > 10000 nM T89697 CVOP58 141744828 IC50 = 450 nM T89697 CC17LW 141744829 IC50 > 10000 nM T89697 CWNS62 141744830 IC50 > 10000 nM T89697 CR5B2L 141744831 IC50 = 950 nM T89697 C8V9BA 141744832 IC50 > 10000 nM T89697 CVK4X8 141744833 IC50 > 10000 nM T89697 CU7VO6 141744834 IC50 = 69 nM T89697 CVF1I5 141744835 IC50 = 680 nM T89697 CYKD76 141744836 IC50 = 90 nM T89697 CEC19U 141744837 IC50 > 10000 nM T89697 C2AT5E 141744838 IC50 > 10000 nM T89697 C9INH5 141744839 IC50 > 10000 nM T89697 CEBS63 141744841 IC50 > 10000 nM T89697 CQMU70 141744842 IC50 > 10000 nM T89697 CW1JR2 141744843 IC50 = 46 nM T89697 C0VD7G 141744844 IC50 > 10000 nM T89697 CL8XN3 141744845 IC50 = 2530 nM T89697 CFP60C 141744846 IC50 > 10000 nM T89697 C96KQW 141744848 IC50 > 10000 nM T89697 CRJ3S0 141744849 IC50 = 530 nM T89697 C0EYH1 142341866 IC50 = 13 nM T89697 C6UAR5 142341947 IC50 = 8.1 nM T89697 CKRU13 142341971 IC50 = 16 nM T89697 CKDT74 142341993 IC50 = 84 nM T89697 CF9N0H 142342024 IC50 = 17 nM T89697 C1JQ0Z 142342046 IC50 = 8.4 nM T89697 CB59EZ 142509480 IC50 = 5.6 nM T89697 C47ERW 142509516 IC50 = 4.3 nM T89697 CTH94V 142509574 IC50 = 21 nM T89697 CZFT65 142509579 IC50 = 66.1 nM T89697 CE9WC7 142509586 IC50 = 16.9 nM T89697 CNQ50X 142509588 IC50 = 4.8 nM T89697 C0S9PQ 142619907 EC50 = 1450 nM T89697 C7JKA2 142619908 EC50 = 10800 nM T89697 CL2AV8 142619909 EC50 = 320 nM T89697 CP1UF7 142619910 EC50 = 6260 nM T89697 CQ8OU6 142619912 EC50 = 4190 nM T89697 C12KDR 142619913 EC50 = 6400 nM T89697 C5H7FG 142619916 EC50 = 6920 nM T89697 CI31ZV 142619918 EC50 = 10700 nM T89697 CM8P4F 142619919 EC50 = 260 nM T89697 CEY1X4 142619920 EC50 = 11000 nM T89697 CH2E7P 142619921 EC50 = 1040 nM T89697 C1CEU5 142619922 EC50 = 18700 nM T89697 CZ9IW2 142619923 IC50 = 1600 nM T89697 CYB27V 142619924 EC50 = 890 nM T89697 C67QGT 142619926 EC50 = 4590 nM T89697 C3LOW2 142619927 EC50 = 5550 nM T89697 CWEC07 142619928 EC50 = 12000 nM T89697 CLU62H 142619929 EC50 = 4560 nM T89697 C5GJ8V 142619931 EC50 = 480 nM T89697 C16SVH 142619932 EC50 = 9120 nM T89697 C9U3KI 142619933 EC50 = 9470 nM T89697 C6NQ9I 145720956 IC50 = 14000 nM T89697 CO40MZ 145951275 EC50 = 5010 nM T89697 C8XCW4 145953593 EC50 = 4290 nM T89697 C5H4UJ 145954041 IC50 = 18 nM T89697 C09ZQS 145954548 IC50 = 1.8 nM T89697 CV6HZ0 145959475 EC50 = 3090 nM T89697 C96GIW 145964069 IC50 = 450 nM T89697 CA7B3R 145964241 IC50 = 200 nM T89697 C9HKR1 145964500 IC50 = 76580 nM T89697 CUA2K5 145964731 IC50 = 580 nM T89697 CT20SR 145965635 IC50 = 60880 nM T89697 CN6SK2 145965768 IC50 = 80580 nM T89697 CK23NR 145966752 IC50 = 5030 nM T89697 CAP6W8 145966837 IC50 = 28 nM T89697 CE5I7C 145967008 IC50 = 65920 nM T89697 CSQJ42 145967348 IC50 = 97 nM T89697 CYN5V8 145967463 IC50 = 58110 nM T89697 CBJ3P1 145967730 IC50 = 2200 nM T89697 C65NHX 145968756 IC50 = 1200 nM T89697 CQ21PR 145968804 IC50 = 4200 nM T89697 C4EZN1 145969081 IC50 = 2200 nM T89697 CPNZ97 145969599 IC50 = 810 nM T89697 CCG1P0 145969967 IC50 = 5700 nM T89697 CLY2T3 145970519 IC50 = 690 nM T89697 C6K9GW 145971318 IC50 = 66730 nM T89697 C2VBX5 145972107 IC50 = 10200 nM T89697 CS5TW7 145973304 IC50 = 82120 nM T89697 CAK60H 145973431 IC50 = 630 nM T89697 CU6KO4 145973699 IC50 = 405 nM T89697 CNV36S 145974038 IC50 = 22730 nM T89697 C0W2XY 145974378 IC50 = 730 nM T89697 CV6Y2O 145976341 IC50 = 20680 nM T89697 CS1O9L 145976459 IC50 = 49340 nM T89697 CSV9N2 145976739 IC50 = 870 nM T89697 CLI94M 145978059 IC50 = 71700 nM T89697 CHWK59 145978347 IC50 = 340 nM T89697 CZW46Y 145978425 IC50 > 1000 nM T89697 CG4M5X 145979054 IC50 = 27 nM T89697 C5SK4O 145979193 IC50 = 209.6 nM T89697 C8CXN2 145979858 EC50 = 480 nM T89697 CRYW71 145980148 IC50 = 2200 nM T89697 C3UG5E 145980172 IC50 = 207.9 nM T89697 CX35HL 145980717 IC50 = 8330 nM T89697 C1IGW2 145980819 IC50 > 100000 nM T89697 CS4MI8 145981708 IC50 = 9500 nM T89697 CW8B6A 145981750 IC50 = 22 nM T89697 C3X8OD 145981785 IC50 = 151.8 nM T89697 CV1RQ9 145981894 EC50 = 330 nM T89697 C7S9MG 145982245 IC50 = 233.7 nM T89697 C2YO8R 145982459 IC50 = 4100 nM T89697 CHT8M1 145982739 IC50 = 87 nM T89697 C9VS3X 145982780 IC50 = 7 nM T89697 CC7ZF9 145982970 IC50 = 394 nM T89697 CHN2M6 145982993 IC50 = 390 nM T89697 CCLP04 145983079 IC50 = 23 nM T89697 C4AKU1 145983122 IC50 = 119 nM T89697 CG02AM 145983180 IC50 = 597.8 nM T89697 C2NH0Y 145983235 IC50 = 39 nM T89697 CPR1W2 145983299 IC50 = 148 nM T89697 CQF57C 145983500 IC50 = 288 nM T89697 C50ZIQ 145984327 IC50 = 448 nM T89697 CH1X5E 145984494 IC50 = 361 nM T89697 C5U2QK 145984896 IC50 = 122.5 nM T89697 CJC34M 145984936 IC50 = 134 nM T89697 C69OSL 145985132 IC50 = 299 nM T89697 C2O7XA 145985324 IC50 = 1192 nM T89697 C4TBS0 145985331 IC50 = 438 nM T89697 CF3ME9 145985603 IC50 = 427 nM T89697 CP09AH 145985633 IC50 > 100000 nM T89697 CKJ8O3 145985919 IC50 = 420 nM T89697 CK0MI7 145985929 IC50 = 50 nM T89697 CM81NX 145986030 IC50 = 117 nM T89697 C3QCS5 145986385 IC50 = 133 nM T89697 CT71UQ 145986568 IC50 = 890 nM T89697 CEJR90 145986692 IC50 = 11000 nM T89697 CJ3TE7 145986756 IC50 = 119.6 nM T89697 C3P0BK 145986889 IC50 = 1100 nM T89697 C05UPF 145987627 IC50 = 18 nM T89697 CGT41S 145987994 EC50 = 460 nM T89697 CH8S9C 145988339 IC50 = 50300 nM T89697 C02ART 145988358 IC50 = 18 nM T89697 CFRN35 145988434 IC50 = 167.9 nM T89697 CDGV74 145988791 IC50 = 1500 nM T89697 CL05NY 145989048 IC50 = 2800 nM T89697 CHJD48 145989519 IC50 = 1580 nM T89697 C29ITB 145989650 IC50 = 338 nM T89697 CI8WB3 145989715 IC50 = 4000 nM T89697 CQ7JU8 145989915 IC50 = 7800 nM T89697 CLK52R 145990092 IC50 = 113.4 nM T89697 CB15WE 145990300 IC50 = 42200 nM T89697 C13KCJ 145990635 IC50 = 2250 nM T89697 CVN6T9 145990888 IC50 = 13590 nM T89697 CKU2L4 145991209 IC50 = 139.8 nM T89697 CX7J2S 145991557 IC50 = 134 nM T89697 CV9DX7 145991568 IC50 = 684 nM T89697 CV61QH 145991788 IC50 = 577.2 nM T89697 CB0ZR4 145992186 IC50 = 3300 nM T89697 C2L0NS 145992195 IC50 = 2700 nM T89697 CJC82P 145993052 IC50 = 61 nM T89697 CYQ79U 145993068 IC50 = 11000 nM T89697 CNWY78 145993645 IC50 = 1950 nM T89697 CR6XN8 145994164 IC50 = 590 nM T89697 CD4WA8 145994224 IC50 = 450 nM T89697 C3SY9B 146018670 IC50 = 16.4 nM T89697 C31MCG 146018671 IC50 = 102.1 nM T89697 C6EF3U 146633829 IC50 = 6.4 nM T89697 C9CH8X 146634682 IC50 = 12.4 nM T89697 C8J3TV 146669430 IC50 = 740 nM T89697 CHE6V5 148026225 IC50 = 12 nM T89697 C1I7JK 148270333 IC50 = 12 nM T89697 C20YQK 153434844 IC50 = 19 nM T89697 CJM43I 153434859 IC50 = 13 nM T89697 C36ISR 153434865 IC50 = 10 nM T89697 CZ7JQ2 153434882 IC50 = 12 nM T89697 C63FMQ 154601093 IC50 = 21 nM T89697 C59HOL 155510561 IC50 > 200 nM T89697 C4JB1R 155511259 IC50 = 70 nM T89697 CF3V7Y 155511297 IC50 = 150 nM T89697 CZT0W5 155511328 IC50 > 1000 nM T89697 CLWA53 155511337 IC50 = 358 nM T89697 C7PTI6 155511361 IC50 = 23000 nM T89697 C6ED7O 155511708 IC50 = 27.6 nM T89697 CX5QS1 155511756 IC50 = 7.6 nM T89697 CWDH25 155511770 IC50 = 18.9 nM T89697 CX04BL 155512330 IC50 = 7200 nM T89697 CHD3C4 155512917 IC50 > 10000 nM T89697 CAG5F0 155513388 IC50 = 1760 nM T89697 CRYM58 155513720 IC50 = 43800 nM T89697 C8VD2I 155513747 IC50 = 781 nM T89697 CHP5L0 155514083 IC50 = 2890 nM T89697 C16XWD 155514212 IC50 = 45.7 nM T89697 CV32TF 155514242 IC50 = 126 nM T89697 CYFW59 155514258 IC50 = 1090 nM T89697 C3CD4X 155514316 IC50 = 3350 nM T89697 CNUW02 155514339 IC50 = 37.2 nM T89697 CX4JQ3 155514783 IC50 = 132 nM T89697 C0G6CR 155515087 IC50 = 14 nM T89697 CES90B 155515098 IC50 = 571 nM T89697 C7LFA0 155515243 IC50 = 457 nM T89697 C1FTN9 155515411 IC50 > 1000 nM T89697 C0H6ZE 155515556 IC50 = 36.9 nM T89697 CCJ14L 155516448 IC50 = 14 nM T89697 CVP8Q5 155516616 IC50 = 16.8 nM T89697 CI4LE2 155516619 IC50 = 28.7 nM T89697 CWJS36 155516630 IC50 = 4.5 nM T89697 CNJ47R 155516651 IC50 = 636 nM T89697 CJ0FH7 155516689 IC50 = 6740 nM T89697 C7IBH0 155516857 IC50 = 657 nM T89697 C4NC7Q 155517508 IC50 = 19.1 nM T89697 CN46XW 155517655 IC50 = 2220 nM T89697 C34RQN 155518507 IC50 = 1094 nM T89697 CJA45U 155518566 IC50 = 1260 nM T89697 CGCO97 155518865 IC50 = 22.2 nM T89697 C9T7MC 155519004 IC50 = 17.9 nM T89697 C8W6QP 155519650 IC50 > 10000 nM T89697 CIW3F0 155519816 IC50 = 72 nM T89697 CO1DT2 155520102 IC50 = 822.5 nM T89697 CH9XP5 155520130 IC50 = 341 nM T89697 C2F6OX 155520170 IC50 = 7150 nM T89697 CZ57XQ 155520612 IC50 = 767 nM T89697 C3ZP5H 155521897 IC50 = 17000 nM T89697 CZ8FN1 155522016 IC50 = 21.4 nM T89697 C4BLS9 155522057 IC50 = 99.4 nM T89697 CTL2I9 155522175 IC50 = 477 nM T89697 C8FS1P 155523075 IC50 = 259 nM T89697 C6B4EL 155523872 IC50 = 24 nM T89697 CRJ9O3 155524304 IC50 = 24 nM T89697 CMDH32 155524514 IC50 = 119 nM T89697 C4PW8J 155524534 IC50 = 14500 nM T89697 CLY12I 155525014 IC50 = 14700 nM T89697 CZK57D 155525299 IC50 = 21 nM T89697 CA01HU 155525338 IC50 = 74.5 nM T89697 CHZD38 155525566 IC50 = 14.4 nM T89697 CY1I6V 155525573 IC50 = 284 nM T89697 CLY5M4 155525580 IC50 = 501.6 nM T89697 CQ3W2E 155525624 IC50 = 3195.3 nM T89697 CC1R5A 155525641 IC50 = 72.9 nM T89697 C3EJR0 155525993 IC50 = 36 nM T89697 C27HXG 155526119 IC50 = 696 nM T89697 C8E5PM 155526671 IC50 = 73.9 nM T89697 CH4KS8 155526712 IC50 = 42 nM T89697 C8TWV7 155527273 IC50 = 338.8 nM T89697 C6VK2Q 155527721 IC50 = 107.4 nM T89697 CCH6I4 155528124 IC50 = 104 nM T89697 C5FW7I 155528311 IC50 = 461 nM T89697 C4LCP3 155528885 IC50 = 44 nM T89697 CA30OB 155529610 IC50 = 44 nM T89697 CZ39JY 155529671 IC50 = 96870 nM T89697 CU3K9S 155529868 IC50 = 94 nM T89697 C13JBA 155530161 IC50 = 148 nM T89697 CYX4D6 155530375 IC50 > 1000 nM T89697 C5X7DV 155530398 IC50 = 35 nM T89697 CYBZ42 155530883 IC50 = 100000 nM T89697 C58PHY 155531191 IC50 = 33 nM T89697 CF5N2S 155531195 IC50 = 3870 nM T89697 CCWU58 155531250 IC50 = 150 nM T89697 CHQ8N5 155531385 IC50 = 2830 nM T89697 CCR71O 155531812 IC50 = 134 nM T89697 C3CVZ1 155532036 IC50 = 73 nM T89697 C5A8MO 155532280 IC50 = 96870 nM T89697 CAQ2Y8 155532641 IC50 = 105000 nM T89697 C3F6ZI 155532803 IC50 = 1281.3 nM T89697 CXS20Z 155532816 IC50 = 418 nM T89697 C70XJB 155533149 IC50 = 21000 nM T89697 CG1K4V 155533289 IC50 = 8000 nM T89697 C7OEH8 155533973 IC50 > 1000 nM T89697 C86BTK 155536043 IC50 = 407 nM T89697 C4H8XB 155536067 IC50 = 20.8 nM T89697 CJVZ35 155536135 IC50 = 10100 nM T89697 C9X7LC 155536325 IC50 = 23 nM T89697 C0O4AQ 155536365 IC50 = 870 nM T89697 CC80FB 155536449 IC50 = 27300 nM T89697 C6RJ2I 155537896 IC50 = 19.2 nM T89697 CXC91A 155538594 IC50 = 817 nM T89697 C0HXA8 155538715 IC50 = 764 nM T89697 CR6EJ3 155539196 IC50 = 25 nM T89697 CFKI70 155539267 IC50 = 10.1 nM T89697 CJ5FY6 155539290 IC50 = 52.7 nM T89697 CR8EP5 155539904 IC50 = 45 nM T89697 CQT17I 155540569 IC50 = 36.3 nM T89697 CJYR81 155540830 IC50 = 29.5 nM T89697 C58KYQ 155540941 IC50 = 2.5 nM T89697 CD3Y5U 155540952 IC50 = 590 nM T89697 CPKO04 155541165 IC50 = 7.4 nM T89697 C4C6RX 155541201 IC50 = 113 nM T89697 CFOQ59 155541414 IC50 = 218.8 nM T89697 CK01YF 155541436 IC50 = 24 nM T89697 C9TJ2I 155541446 IC50 = 112 nM T89697 CP5R8Z 155541668 IC50 = 850 nM T89697 CF3AW0 155541799 IC50 = 1730 nM T89697 CP25JB 155542022 IC50 = 151 nM T89697 CLC81R 155542366 IC50 = 8.7 nM T89697 C02NAK 155542721 IC50 = 691 nM T89697 C94KJF 155543368 IC50 = 217 nM T89697 CKN39Q 155544466 IC50 = 399 nM T89697 CIUK86 155544692 IC50 = 26 nM T89697 CI9O0P 155544755 IC50 = 143 nM T89697 CZAL46 155545224 IC50 = 9 nM T89697 C1Z5EA 155545364 IC50 = 44.9 nM T89697 CHN82B 155546259 IC50 > 1000 nM T89697 CNPU01 155546283 IC50 = 2741 nM T89697 CE04JU 155546342 IC50 = 327 nM T89697 C0OC8M 155547213 IC50 = 322 nM T89697 C0C8FP 155547279 IC50 = 9.6 nM T89697 CN03BT 155547734 IC50 = 7.1 nM T89697 CMH35W 155547809 IC50 = 3.3 nM T89697 CWX19H 155548140 IC50 = 6.6 nM T89697 C9J2RI 155548653 IC50 = 306 nM T89697 C8C3SW 155548933 IC50 = 180 nM T89697 CYD57L 155549229 IC50 > 1000 nM T89697 CGZ2A8 155549756 IC50 = 539 nM T89697 C3NX1M 155549772 IC50 > 200 nM T89697 CH96DK 155550037 IC50 = 2480 nM T89697 C6O7LQ 155550877 IC50 > 10000 nM T89697 C2GSR8 155550907 IC50 = 969 nM T89697 C6JV3E 155551216 EC50 = 690 nM T89697 CSU75P 155551311 IC50 = 22 nM T89697 CNU93S 155551336 IC50 = 7.8 nM T89697 C20NJG 155551633 IC50 = 73.2 nM T89697 C3YG1T 155551998 EC50 = 4200 nM T89697 CX5NG6 155552179 IC50 = 51.7 nM T89697 CN46IF 155552796 IC50 = 35.7 nM T89697 CE95UF 155552938 IC50 = 3360 nM T89697 C8M1QG 155553198 IC50 = 939 nM T89697 C0ASJ7 155553201 EC50 = 2600 nM T89697 C12IJV 155553541 EC50 = 24000 nM T89697 C20SOV 155554077 IC50 > 10000 nM T89697 CQ7BU3 155554221 IC50 = 5.7 nM T89697 C6U9KC 155555102 IC50 = 7153.3 nM T89697 CQ6D7M 155555581 IC50 = 19 nM T89697 C6HNU8 155555675 IC50 = 102 nM T89697 C6DKG1 155555719 IC50 = 75 nM T89697 C86QJW 155556390 IC50 = 10.5 nM T89697 CA3KH1 155556529 IC50 = 4.6 nM T89697 C63AHT 155557140 IC50 > 1000 nM T89697 C0XC9H 155557271 IC50 = 223 nM T89697 CO7P3Z 155557740 IC50 = 933 nM T89697 CI0V8G 155558434 IC50 = 1072.1 nM T89697 C4RWF1 155558731 IC50 = 27 nM T89697 C1TIH7 155558824 IC50 = 33 nM T89697 C5QB1Y 155558872 IC50 = 304 nM T89697 CBYL12 155559016 IC50 = 1910 nM T89697 CU8L5V 155559057 IC50 = 4 nM T89697 CJ82RN 155559113 IC50 = 55.8 nM T89697 CZ14NM 155559275 EC50 = 340 nM T89697 CNJ4C7 155559429 IC50 > 1000 nM T89697 CQY4A1 155560339 IC50 = 743.9 nM T89697 CA48WP 155560350 IC50 = 24000 nM T89697 C6R2SJ 155560411 IC50 = 58350 nM T89697 C7ZPV4 155560705 IC50 = 354 nM T89697 CQIT48 155560791 IC50 = 3814 nM T89697 CQT16B 155561274 IC50 = 14.6 nM T89697 CEK9J1 155561942 IC50 = 10.1 nM T89697 C25KBO 155562131 IC50 = 357 nM T89697 CFX43K 155562566 IC50 = 19 nM T89697 C3NDJ2 155562711 IC50 = 1090 nM T89697 CSQ8U0 155562797 IC50 = 2734 nM T89697 CF5G4Y 155563108 IC50 > 200 nM T89697 CB4E0U 155563312 IC50 = 38.1 nM T89697 CC7P0V 155563603 IC50 = 20.3 nM T89697 CXMP83 155564029 IC50 > 1000 nM T89697 C4MJ7U 155564599 IC50 = 19.5 nM T89697 CG02FV 155564613 IC50 = 1990 nM T89697 C2C7EU 155564852 IC50 = 255.5 nM T89697 CP19JR 155564990 IC50 = 8.5 nM T89697 CXM8P9 155565017 IC50 = 1020 nM T89697 C83WCP 155565053 IC50 > 1000 nM T89697 CG43BS 155565222 IC50 = 2200 nM T89697 CFP34M 155565482 IC50 = 5623 nM T89697 CP5Y9H 155566146 IC50 = 110000 nM T89697 CNX9T1 155566545 IC50 = 138 nM T89697 CY5LV8 155566655 IC50 = 7.5 nM T89697 CEA02R 155566797 IC50 = 37.1 nM T89697 C61SEH 155567075 IC50 = 1210 nM T89697 CFN2U7 155567243 IC50 = 413 nM T89697 CN91VH 155567244 IC50 = 221 nM T89697 CI0D1N 155567338 IC50 = 855 nM T89697 C07ASO 155567542 IC50 = 3563 nM T89697 CO58ME 155567694 EC50 = 10000 nM T89697 CB19FR 155567818 IC50 = 62.5 nM T89697 C2O8RC 155568012 IC50 = 1430 nM T89697 CW45BT 155568279 IC50 = 4.2 nM T89697 CAH57R 155569047 IC50 > 10000 nM T89697 C6OA1Z 155569140 IC50 = 258 nM T89697 CU3Y0S 155569235 IC50 = 5.1 nM T89697 CSB45Q 155569293 EC50 = 670 nM T89697 D00BGN 24971326 IC50 = 5300 nM T89697 D00GYX 7509 IC50 = 1700 nM T89697 D00UIK 17937479 IC50 = 2500 nM T89697 D00XOT 45487214 IC50 = 12500 nM T89697 D01CSZ 44466195 IC50 = 15000 nM T89697 D01HST 1085108 IC50 = 3000 nM T89697 D02ADV 594397 IC50 = 1000000 nM T89697 D02DRL 199161 IC50 = 4800 nM T89697 D02IVJ 2803022 IC50 = 2000 nM T89697 D02SRL 3000729 IC50 = 4000 nM T89697 D02XRG 45487209 IC50 = 50000 nM T89697 D03ETX 44406807 Ki = 13220 nM T89697 D03JAE 12465608 IC50 = 800 nM T89697 D03JMD 49866094 IC50 = 2600 nM T89697 D04OXY 16871 IC50 = 720 nM T89697 D05AFW 49866090 IC50 = 16000 nM T89697 D05LFV 12526770 IC50 = 6800 nM T89697 D06MUL 44406804 Ki = 17150 nM T89697 D06OUR 44466196 IC50 = 3000 nM T89697 D06YFT 676159 IC50 = 78 nM T89697 D07NSZ 13266247 IC50 = 1400 nM T89697 D07NYX 7222 IC50 = 652000 nM T89697 D08GZK 24856337 Ki = 80 nM T89697 D08MOG 45487171 IC50 = 3500 nM T89697 D08MRL 45487219 IC50 = 4500 nM T89697 D08PIF 80407 IC50 = 1400 nM T89697 D08XXD 17815 IC50 = 6000 nM T89697 D08YGW 10444038 IC50 = 32000 nM T89697 D08YHA 72734 IC50 = 214 nM T89697 D09BVH 11305 IC50 = 10000 nM T89697 D09DSZ 3266369 IC50 = 7000 nM T89697 D09JOM 15945669 IC50 = 400 nM T89697 D09ZJW 80409 IC50 = 1100 nM T89697 D0A7NH 45487176 IC50 = 15000 nM T89697 D0B9IA 16091658 Ki = 140 nM T89697 D0DB2N 16059787 Ki = 690 nM T89697 D0DQ6Z 8530 IC50 = 460 nM T89697 D0FO2B 1923 IC50 = 750000 nM T89697 D0G0EE 24971327 Ki = 5300 nM T89697 D0G8IH 20029042 IC50 = 12500 nM T89697 D0GJ7J 3760 IC50 = 23000 nM T89697 D0H0HM 135411931 IC50 = 2560 nM T89697 D0I2RW 8342 IC50 = 280 nM T89697 D0I9AT 73549 IC50 = 53.7 nM T89697 D0J9DD 69590 Ki = 4400 nM T89697 D0K3SZ 78252 IC50 = 1300 nM T89697 D0K4MG 21609882 Ki = 2300 nM T89697 D0MC4U 16066751 Ki = 41 nM T89697 D0N1ZJ 44465947 IC50 = 4000 nM T89697 D0NI8W 10307884 IC50 = 1200 nM T89697 D0O3IE 137153 IC50 = 8900 nM T89697 D0O9QG 68342 IC50 = 2200 nM T89697 D0P1CO 2830968 IC50 = 7300 nM T89697 D0P3XW 580759 IC50 = 1200 nM T89697 D0PR7L 85171 IC50 = 1800 nM T89697 D0Q9JG 13885856 IC50 = 10000 nM T89697 D0R6FJ 64961 Ki = 120 nM T89697 D0S1FF 44465702 IC50 = 2500 nM T89697 D0SZ9F 95756 IC50 = 3500 nM T89697 D0TM0Z 152300 Ki = 190 nM T89697 D0UV8T 9942176 IC50 = 5000 nM T89697 D0V8FG 81062 IC50 = 320000 nM T89697 D0W3ON 416002 IC50 = 3000 nM T89697 D0W3OY 78062 IC50 = 2200 nM T89697 D0W3XP 356405 Ki = 1200 nM T89697 D0W9VA 10667 IC50 = 7100 nM T89697 D0Z0BB 118986 IC50 = 100 nM T89697 D0Z3NE 478573 IC50 = 0.018 nM T89697 D0Z4JG 11074644 IC50 = 5500 nM T22977 CSTX48 12029908 IC50 = 381100 nM T22977 CFCQ32 24823795 IC50 = 365800 nM T22977 CCM1W9 24823796 IC50 = 67900 nM T22977 C78RBD 24823798 IC50 = 786900 nM T22977 CV75UN 24823942 IC50 = 129300 nM T22977 CFG3S8 24970402 IC50 = 56600 nM T22977 CU16PV 34363640 EC50 = 1930 nM T22977 CGCZ64 45102767 EC50 = 67 nM T22977 C0ZCI8 46196578 EC50 = 790 nM T22977 C1S4FQ 46215250 EC50 > 32000 nM T22977 C10GXV 46215251 EC50 = 1470 nM T22977 C2P4ZD 46215255 EC50 = 4700 nM T22977 CUMR17 50993705 EC50 = 170 nM T22977 CD49KF 51003102 IC50 = 96600 nM T22977 CB50PY 51003103 IC50 = 103300 nM T22977 CUQ4H3 53324606 EC50 = 710 nM T22977 C9V4XG 56945435 EC50 = 2880 nM T22977 CPDZ84 56945436 EC50 = 1410 nM T22977 C0Y8TI 56945437 EC50 = 1960 nM T22977 C4YE3U 56945438 EC50 = 720 nM T22977 CBLU36 56945439 EC50 = 870 nM T22977 CM40FZ 56945440 EC50 = 580 nM T22977 C0ZL2B 56945548 EC50 = 1070 nM T22977 CMRJ61 56945549 EC50 = 510 nM T22977 CTGZ70 56945550 EC50 = 1020 nM T22977 C4TK9D 56945551 EC50 = 2840 nM T22977 C0XJU1 56945552 EC50 = 3700 nM T22977 CPB16S 62140981 IC50 = 83120 nM T22977 CS43AO 71459115 IC50 = 71460 nM T22977 CTWB85 71460923 IC50 = 125320 nM T22977 COD7K9 71462627 IC50 = 65980 nM T22977 C2DM8H 71652393 IC50 = 408000 nM T22977 CL7I0C 71652552 IC50 = 178500 nM T22977 C81MVZ 71652554 IC50 = 641000 nM T22977 C47ETO 101519736 IC50 = 58900 nM T22977 CKI9V6 145960712 IC50 > 100000 nM T22977 CQ2D5R 145961082 IC50 = 100000 nM T22977 C6AX9C 145963675 IC50 = 145800 nM T22977 CW2LP6 155518910 IC50 > 100000 nM T22977 C5D3QO 155521025 IC50 > 100000 nM T22977 CQM2B3 155521222 IC50 > 100000 nM T22977 CABH43 155522156 IC50 > 100000 nM T22977 CNH43F 155533839 IC50 > 50000 nM T22977 C8H4CG 155537441 IC50 > 50000 nM T10756 C06BAM 219561 IC50 = 8900 nM T10756 CV5HI2 219565 IC50 = 11000 nM T10756 C8ZR3J 256755 IC50 = 8800 nM T10756 CFWY79 10099159 IC50 = 7000 nM T10756 C3YE9J 10393519 IC50 = 7000 nM T10756 C0QT1V 11758430 IC50 = 14000 nM T10756 CLG8I5 44178850 IC50 > 100 ug.mL-1 T10756 C94LUQ 44178851 IC50 = 38 ug.mL-1 T10756 CN84ZR 45270893 IC50 = 9 ug.mL-1 T10756 C3Z4TA 45271732 IC50 = 4.2 ug.mL-1 T10756 C2W3DX 127038789 IC50 = 5000 nM T10756 CP3W5G 127038790 IC50 = 4200 nM T10756 C6UQ9T 127038791 IC50 = 5300 nM T10756 CX2U4F 127039115 IC50 = 3900 nM T10756 C04WTC 127039117 IC50 = 5400 nM T10756 C08HWM 127040772 IC50 = 14000 nM T10756 CCE90R 127040773 IC50 = 9800 nM T10756 CUST62 127041091 IC50 = 16000 nM T10756 CJ2U3N 127041092 IC50 = 7100 nM T10756 CREI95 127041093 IC50 = 6700 nM T10756 C7UI6S 127041094 IC50 = 8200 nM T10756 CK1Q6H 127041986 IC50 = 38000 nM T10756 C93YZB 127042064 IC50 = 9400 nM T10756 C0AR9E 127042065 IC50 = 3800 nM T10756 C62BOX 127042391 IC50 = 4900 nM T10756 D0F3TM 219564 IC50 = 6900 nM T41702 D0E3TC 44259 IC50 = 7440 nM T41702 CEC30Q 3674 IC50 > 40000 nM T41702 CN64JR 8323 IC50 = 26200 nM T41702 C3YRU7 15295578 IC50 = 250 nM T41702 C2UOE0 24766030 IC50 > 50000 nM T41702 CY8L7E 24896769 IC50 > 10000 nM T41702 CLFM35 25206064 IC50 = 520 nM T41702 CK73NR 44219749 IC50 > 50000 nM T41702 C3VRO9 44557921 IC50 = 9549.93 nM T41702 CCL85F 44575073 IC50 > 50000 nM T41702 CJX06P 44575126 IC50 = 4900 nM T41702 CE8FC7 44575127 IC50 = 11600 nM T41702 C28QLM 44605035 IC50 = 17900 nM T41702 C75XHS 44605037 IC50 > 50000 nM T41702 CC95PQ 45375865 IC50 > 50000 nM T41702 CEOQ27 45375866 IC50 > 50000 nM T41702 C96BNW 46179972 IC50 > 50000 nM T41702 CO3P0J 46866604 IC50 < 50000 nM T41702 CLS29B 46872626 IC50 > 10000 nM T41702 CJOM49 46880136 IC50 = 9510 nM T41702 CV63UL 67240318 IC50 > 10000 nM T41702 C2MD1Q 155513187 IC50 > 10000 nM T41702 D01YWE 25207521 IC50 = 160 nM T41702 D0L4WN 31420 IC50 = 34000 nM T41702 D0Y6OK 6688 IC50 > 40000 nM T89041 D00AXJ 4189 Ki = 243 nM T89041 D02STN 132971 IC50 ~ 1 nM T89041 D06CNP 9821849 IC50 = 18 nM T89041 D07ABV 468595 IC50 = 42 nM T89041 D09GOS 2812 Ki = 81.5 nM T89041 D09LNI 3365 IC50 > 200000 nM T89041 D0AA2D 2378 Ki = 56.5 nM T89041 D0B4IF 456201 IC50 = 1800 nM T89041 D0CA6J 5482 Ki = 505 nM T89041 D0EV8E 3198 Ki = 325 nM T89041 D0M6DO 2145 IC50 = 60000 nM T89041 D0Q9JT 4174 IC50 > 10000 nM T89041 D0ZX1P 59693 IC50 > 5000 nM T89041 D03AJU 44139752 IC50 = 3981.07 nM T89041 D0U0BU 11188409 IC50 = 28.1 nM T89041 D0X3OI 9883029 IC50 = 38 nM T89041 D0SX7F 60876 Ki = 447 nM T89041 C9LCD8 3823 IC50 = 26 nM T89041 CWMQ17 92747 IC50 = 1430 nM T89041 C8EQ1Z 92855 IC50 = 1710 nM T89041 C2GRN7 94199 IC50 = 440 nM T89041 C7VP8E 101966 IC50 = 800 nM T89041 CHWM72 125921 IC50 > 34000 nM T89041 CYSE03 196941 IC50 = 6.13 nM T89041 CUP91R 245872 IC50 = 66 nM T89041 CPE17Q 320374 IC50 = 43900 nM T89041 C7TYH9 585624 IC50 = 18000 nM T89041 CUL8N9 709713 IC50 > 31622.78 nM T89041 C3H1DE 2998104 IC50 = 1600 nM T89041 C1WIR4 4499193 IC50 > 31622.78 nM T89041 CA15IT 9796590 IC50 = 19 nM T89041 CC3QF5 9797875 Ki = 1.9 nM T89041 C9QVL1 9816909 IC50 = 130 nM T89041 C9D4MI 9819290 Ki = 1.4 nM T89041 CRQA29 9830290 IC50 = 28 nM T89041 CKJ1I6 9838340 IC50 = 18 nM T89041 CBZQ79 9840765 Ki = 41 nM T89041 CN9U6I 9840821 Ki = 1.2 nM T89041 CAQ52K 9861918 IC50 = 15 nM T89041 CL2W9Z 9862746 Ki = 1.4 nM T89041 CUK64X 9880846 IC50 = 400 nM T89041 CQHE82 9883170 IC50 = 19 nM T89041 C8YQ6V 9883171 IC50 = 27 nM T89041 C5VA7T 9884336 Ki = 23 nM T89041 CJ56EL 9904146 IC50 = 18 nM T89041 CG0I7C 9905837 IC50 = 39 nM T89041 CUZT98 9906455 IC50 = 75 nM T89041 C4PF5A 9923132 IC50 = 190 nM T89041 CWL3O1 9926844 IC50 = 75 nM T89041 C3TH4Q 9927224 IC50 = 16 nM T89041 C7LSP1 9927786 Ki = 8 nM T89041 C8RPF6 9949067 IC50 = 130 nM T89041 C3IQV6 9965885 IC50 = 29 nM T89041 CO1Z0A 9971194 IC50 = 1.8 nM T89041 CE3L8V 10061454 IC50 = 1100 nM T89041 CG24IZ 10247264 IC50 = 270 nM T89041 CEMU16 10335364 IC50 = 48 nM T89041 C1OA8L 10337109 IC50 = 50 nM T89041 CB7RI8 10358293 IC50 = 490 nM T89041 C5IZ0X 10380012 IC50 = 13 nM T89041 CR0O6C 10447478 IC50 = 2.7 nM T89041 CQWX01 10450499 IC50 = 1000 nM T89041 C3YI0N 10467502 IC50 = 110 nM T89041 C1JC9V 10521065 IC50 = 108 nM T89041 C86HTI 10522113 IC50 = 400 nM T89041 CFK2N9 10543224 IC50 = 970 nM T89041 C4L8OX 10566080 IC50 = 92 nM T89041 CB90LV 10593280 IC50 = 62 nM T89041 C72XUK 10594248 IC50 = 74 nM T89041 C38SOM 10595962 IC50 = 75 nM T89041 C3OY0Q 10636825 IC50 = 820 nM T89041 C3WZ7D 10638951 Ki = 3 nM T89041 C38WKE 10642746 IC50 = 260 nM T89041 C9QN4J 10660816 IC50 = 150 nM T89041 C82HFM 10663232 IC50 = 1250 nM T89041 C0N2BV 10684551 IC50 = 35 nM T89041 C01ZPW 10684552 IC50 = 320 nM T89041 CPS30O 10689427 IC50 = 5 nM T89041 C7U3ZR 10755577 IC50 = 230 nM T89041 CH8T4Y 10758923 IC50 = 2500 nM T89041 C45HMW 10758924 IC50 > 2500 nM T89041 C3AJ4U 10759395 Ki = 8 nM T89041 CIKB07 10806964 IC50 = 21 nM T89041 C94PCN 10826001 IC50 = 460 nM T89041 CN7I8H 10827014 IC50 = 74 nM T89041 CZW6V4 10828130 IC50 = 220 nM T89041 CE23TU 10831118 IC50 = 219 nM T89041 CY34VS 10854385 Ki = 1.9 nM T89041 C58ETU 11002256 Ki = 1.2 nM T89041 CCFU47 11440648 IC50 = 300 nM T89041 CN4T0K 11544009 IC50 = 233 nM T89041 CZ50DQ 11708478 IC50 = 721 nM T89041 CZH43C 11725276 IC50 = 3 nM T89041 C3N4FE 11792279 IC50 = 27 nM T89041 CHLB06 11855878 IC50 = 1250 nM T89041 C96DPL 11855879 IC50 = 915 nM T89041 C7EF1B 11855880 IC50 = 5817.4 nM T89041 C0EPD3 12039019 IC50 = 220 nM T89041 C13GAW 12043371 IC50 = 54 nM T89041 CZJ0B5 12043372 IC50 = 33 nM T89041 C85ZFQ 12043374 IC50 = 28 nM T89041 CF28CA 12074093 IC50 = 22 nM T89041 CJY17R 12074102 IC50 = 36 nM T89041 CJV5G1 12074103 IC50 = 19 nM T89041 CXQI20 12310542 IC50 = 8000 nM T89041 CLSM38 14872624 IC50 = 140000 nM T89041 C39MVQ 15462429 Ki = 23 nM T89041 CC9BE5 17963726 IC50 = 39 nM T89041 CRL9N5 18395624 IC50 = 42 nM T89041 CX6L9A 18395626 IC50 = 24 nM T89041 CK2AJ8 18668528 IC50 = 49 nM T89041 CI3HL4 18668538 IC50 = 40 nM T89041 CCWH59 18668580 IC50 = 36 nM T89041 CW8PF5 18668583 IC50 = 120 nM T89041 C6ADH5 18668593 IC50 = 24 nM T89041 C4-JAN-02 18668607 IC50 = 45 nM T89041 C9V4BO 18668614 IC50 = 44 nM T89041 CY1HK4 18668617 IC50 = 38 nM T89041 CTA76E 18769059 IC50 = 39 nM T89041 C7UKI6 18769065 IC50 = 200 nM T89041 C0LCW3 18769074 IC50 = 160 nM T89041 C8QA0F 18769127 IC50 = 30 nM T89041 CM9NU7 21852976 IC50 = 3950 nM T89041 CKV94G 21879620 IC50 = 13 nM T89041 C2KMV5 21879624 IC50 = 290 nM T89041 C3DT1N 22018410 IC50 = 28 nM T89041 CXMA20 22018425 IC50 = 36 nM T89041 CT24BF 22664964 IC50 = 24 nM T89041 C0F4YM 22737877 IC50 = 46 nM T89041 CZ2BC5 23288050 IC50 = 40 nM T89041 C59VCE 23424811 IC50 = 2880 nM T89041 C5BVZ6 25022443 IC50 = 345 nM T89041 C29WQM 25033651 IC50 > 10000 nM T89041 C1VPF8 25033652 IC50 = 423 nM T89041 CDR34P 25033653 IC50 = 2346 nM T89041 CE0L8C 25033655 IC50 > 5000 nM T89041 C9Q8ZK 25033657 IC50 > 5000 nM T89041 CWIC10 25033659 IC50 = 307 nM T89041 C32QBZ 25033661 IC50 > 20000 nM T89041 CAI47X 25033725 IC50 = 163 nM T89041 C1XW6O 25033727 IC50 = 144 nM T89041 C23EWR 25033729 IC50 > 20000 nM T89041 CW5A1U 25033730 IC50 = 587 nM T89041 CV49HP 25033731 IC50 > 5000 nM T89041 CJHY97 25033732 IC50 > 20000 nM T89041 C86AIT 25033734 IC50 > 5000 nM T89041 CEJ89P 25033804 IC50 = 188 nM T89041 C3UF1V 25033806 IC50 = 233 nM T89041 CF46OB 25033808 IC50 = 1222 nM T89041 CBI59C 25033810 IC50 = 64 nM T89041 CZPW03 25034656 IC50 > 20000 nM T89041 C7KAR1 25034657 IC50 = 333 nM T89041 CZX08M 25142015 Ki = 54 nM T89041 C0XHA2 25180109 IC50 = 316.23 nM T89041 C1HYO5 40513267 IC50 = 430 nM T89041 CV3Y2B 42642720 IC50 = 90 nM T89041 C9AQ7N 42642721 IC50 = 52 nM T89041 C6GR3F 42642761 IC50 = 379 nM T89041 CQ5M2Z 42642929 IC50 = 261 nM T89041 C2D1MN 42642930 IC50 = 217 nM T89041 CD4OQ8 42643273 IC50 > 5000 nM T89041 CO7YV0 42643327 IC50 = 188 nM T89041 C6UR8G 44315168 IC50 = 3810 nM T89041 C4F5JS 44315175 IC50 = 562 nM T89041 C0B2KL 44315318 IC50 = 1400 nM T89041 C9OPM6 44315319 IC50 = 2600 nM T89041 CO1N3V 44315442 IC50 = 3700 nM T89041 CYKB02 44315468 IC50 = 660.25 nM T89041 C0A4LF 44315469 IC50 = 178.2 nM T89041 CD4VR0 44315540 IC50 = 616.5 nM T89041 CM0ZU4 44315606 IC50 = 225 nM T89041 CY76KC 44315613 IC50 = 500 nM T89041 C5SN0H 44340248 IC50 = 59 nM T89041 CC2E3X 44340275 IC50 = 400 nM T89041 C4PJ1H 44340350 IC50 = 58 nM T89041 CA6B2U 44340378 IC50 = 400 nM T89041 CRW68V 44340379 IC50 = 1113 nM T89041 C5HZX0 44340405 IC50 = 150 nM T89041 CN2DW3 44340421 IC50 = 150 nM T89041 CEGT92 44340434 IC50 > 30000 nM T89041 CECD15 44340462 IC50 = 400 nM T89041 CX9HV5 44340476 IC50 = 1200 nM T89041 CM6PF7 44340585 IC50 = 400 nM T89041 CJ0DG8 44340586 IC50 = 150 nM T89041 C03ATJ 44340924 IC50 = 150 nM T89041 C03EXH 44340925 IC50 = 150 nM T89041 CO8XJ3 44354706 IC50 = 5 nM T89041 C7YDP6 44354757 IC50 = 6 nM T89041 C1W6IR 44354758 IC50 = 9 nM T89041 C4AXM5 44354773 IC50 = 270 nM T89041 CZN1X8 44354907 IC50 = 15 nM T89041 CN8M5U 44354930 IC50 = 88 nM T89041 CCA28Y 44354942 IC50 = 35 nM T89041 CNRO38 44354943 IC50 = 10 nM T89041 CQIP34 44354944 IC50 = 670 nM T89041 CO1W4F 44355172 IC50 = 14 nM T89041 CX2R3P 44355187 IC50 > 1000 nM T89041 CCF7G1 44355188 IC50 = 38 nM T89041 CD4S9E 44357420 IC50 = 1770 nM T89041 CKO6B3 44357421 IC50 = 240 nM T89041 CL2I0F 44357429 IC50 = 510 nM T89041 CZ5VG2 44357431 IC50 = 6480 nM T89041 CU1BG7 44357482 IC50 = 35000 nM T89041 C2WAV8 44357582 IC50 = 720 nM T89041 CJ06LT 44357609 IC50 = 230 nM T89041 C6EY7I 44357615 IC50 = 750 nM T89041 CCN6B1 44357617 IC50 = 890 nM T89041 CO1F8W 44357623 IC50 = 190 nM T89041 CJE4I1 44357624 IC50 = 750 nM T89041 CLZM23 44358638 IC50 > 2500 nM T89041 C64IWU 44358640 Ki = 6 nM T89041 C0SX7B 44358689 IC50 > 25000 nM T89041 CJM80V 44358932 IC50 = 1800 nM T89041 CV5HF6 44367009 IC50 = 27 nM T89041 C4D7ZY 44456181 IC50 = 263 nM T89041 C8VI7P 44456221 IC50 = 236 nM T89041 C6JHB5 44456224 IC50 = 584 nM T89041 C1E8RI 44461114 IC50 = 2.9 nM T89041 CIM9D1 44461115 IC50 > 10000 nM T89041 CQ8MP7 44461136 IC50 = 5.6 nM T89041 C5VF2C 44461174 IC50 = 23 nM T89041 C6RV0L 44461240 IC50 = 160 nM T89041 CY7OD4 44461241 IC50 = 3 nM T89041 CECX12 44461375 IC50 > 10000 nM T89041 CAW3I8 44461376 IC50 = 1.8 nM T89041 CK58SI 44461377 IC50 = 2.5 nM T89041 C2QVD9 44586763 IC50 = 2200 nM T89041 C31AFB 44586764 IC50 = 1700 nM T89041 C1A6IL 44586765 IC50 > 5000 nM T89041 C1TFP5 44586766 IC50 = 3800 nM T89041 CB30QW 44586793 IC50 = 1300 nM T89041 CT38XH 44586824 IC50 > 5000 nM T89041 C4VU2E 44586825 IC50 = 756 nM T89041 CYR4O7 44586826 IC50 > 5000 nM T89041 CH0Y5Z 44586865 IC50 = 168 nM T89041 C7W9EK 44586866 IC50 = 118 nM T89041 CUCM51 44587269 IC50 = 460 nM T89041 CIU9Z3 44587270 IC50 = 1050 nM T89041 C1M6TX 44587293 IC50 > 5000 nM T89041 CH28TE 44587294 IC50 > 5000 nM T89041 CNOG06 44587313 IC50 = 670 nM T89041 C6JSU2 44587318 IC50 = 3100 nM T89041 C7Q6UK 44587319 IC50 > 5000 nM T89041 COM7P5 44587320 IC50 > 5000 nM T89041 C24XTP 44587322 IC50 > 5000 nM T89041 CWF4V8 44587323 IC50 > 5000 nM T89041 CUV83E 46854605 IC50 = 56 nM T89041 CIA08B 46854608 IC50 = 37 nM T89041 C3NO7G 46854609 IC50 = 1458 nM T89041 C0NIH6 46854610 IC50 = 493 nM T89041 C78THB 46854611 IC50 = 852 nM T89041 COVL29 46854757 IC50 > 10000 nM T89041 CWJ3F1 46854758 IC50 = 38 nM T89041 CKRQ67 46854759 IC50 = 75 nM T89041 CZ1YJ0 46854760 IC50 = 62 nM T89041 C9UO5G 46901439 IC50 > 5000 nM T89041 C8LQX7 46901612 IC50 > 5000 nM T89041 CN5G2X 46901617 IC50 = 3340 nM T89041 CC25UL 46901778 IC50 = 1370 nM T89041 C7Y0PC 46901779 IC50 > 10000 nM T89041 CHNF30 46901780 IC50 > 10000 nM T89041 CIC9S5 49799473 IC50 = 75 nM T89041 C9W8HK 49863993 IC50 > 10000 nM T89041 CYMO96 49864179 IC50 > 5000 nM T89041 CNBU93 50994740 IC50 = 19 nM T89041 C6RD7G 53249084 IC50 = 26 nM T89041 CP31IL 53319749 IC50 = 38 nM T89041 C6HPO5 53323744 IC50 = 270 nM T89041 CAE25J 53763992 IC50 = 15 nM T89041 C60LIJ 54580449 IC50 = 22 nM T89041 C8V9GW 54582428 IC50 = 150 nM T89041 C7LHV1 54583409 IC50 = 21 nM T89041 CAO9B4 54584364 IC50 = 77 nM T89041 CAK7Z9 54585325 IC50 = 160 nM T89041 CS51ZD 54585326 IC50 = 340 nM T89041 CSV1M4 54586281 IC50 = 26 nM T89041 C01JOU 54586320 IC50 = 92 nM T89041 C9FBH0 54586321 IC50 = 240 nM T89041 C4N0WL 56645363 IC50 > 10000 nM T89041 C57NSZ 56645568 IC50 > 10000 nM T89041 C6PUX9 56645570 IC50 > 10000 nM T89041 CTW6K2 56645571 IC50 > 10000 nM T89041 CA3VO0 56949328 IC50 = 19 nM T89041 CBMY17 56952125 IC50 = 8 nM T89041 C4EPA7 56952126 IC50 = 37 nM T89041 CDL64H 56952128 IC50 = 396 nM T89041 CX1TL3 56952129 IC50 = 361 nM T89041 C7ND1A 56952239 IC50 = 674 nM T89041 CD94CU 56952242 IC50 = 797 nM T89041 C4R3KU 56952244 IC50 = 135 nM T89041 CNXD75 56952346 IC50 = 330 nM T89041 CQ0IA7 56952348 IC50 = 405 nM T89041 CIO9C5 56953325 IC50 = 8 nM T89041 CEW8L6 56953509 IC50 = 656 nM T89041 C4B1EA 56953512 IC50 = 758 nM T89041 CZG03U 56953601 IC50 = 11 nM T89041 CB1FO5 56953605 IC50 = 40 nM T89041 CONW20 56953606 IC50 = 5.8 nM T89041 C1K2YU 56968076 IC50 = 180 nM T89041 C6ATQ0 57390715 IC50 = 88 nM T89041 CD7M5V 57397795 IC50 = 410 nM T89041 CY97BO 57402969 IC50 = 5.5 nM T89041 C2TUJ7 58255382 IC50 = 2880 nM T89041 C3DPC0 58255407 IC50 > 5000 nM T89041 C9DK1X 58255415 IC50 > 10000 nM T89041 CRQ70M 58255438 IC50 = 1550 nM T89041 CP6RA9 58255482 IC50 > 10000 nM T89041 CW71EO 58255581 IC50 > 10000 nM T89041 CB7N8A 60195126 IC50 > 5000 nM T89041 CX4N0I 62707515 IC50 > 10000 nM T89041 C0G3LA 66559847 IC50 > 10000 nM T89041 C4RSI6 66559935 IC50 > 10000 nM T89041 CDX7I8 66559936 IC50 > 10000 nM T89041 CF9EQ5 66559939 IC50 > 10000 nM T89041 CQN6D3 66559940 IC50 > 10000 nM T89041 CN4H8G 66559941 IC50 > 10000 nM T89041 CTP6Q4 66559942 IC50 > 10000 nM T89041 C9EGW2 66575742 IC50 > 10000 nM T89041 CMXA10 66575743 IC50 > 10000 nM T89041 CKWB91 66575744 IC50 > 10000 nM T89041 C7I3MW 66575745 IC50 > 10000 nM T89041 CPN17S 66575746 IC50 > 10000 nM T89041 CG0ZA7 66575747 IC50 > 10000 nM T89041 C6HF0U 66575748 IC50 > 10000 nM T89041 CDI93T 66575817 IC50 > 10000 nM T89041 CBP6I7 66576773 IC50 > 10000 nM T89041 C4NYB0 66576930 IC50 > 10000 nM T89041 C3LP5H 66576931 IC50 > 10000 nM T89041 CE03WG 66576932 IC50 > 10000 nM T89041 C9DP3R 66850314 IC50 = 25900 nM T89041 C97BGW 69093249 IC50 = 940 nM T89041 CZC4E1 69093450 IC50 = 170 nM T89041 C7ZX9P 69281312 IC50 = 570 nM T89041 C7PY1Q 69281314 IC50 = 74 nM T89041 C1VMF2 70977969 IC50 > 10000 nM T89041 CLR3Q2 71452704 IC50 = 280 nM T89041 CI6B9U 71454429 Ki = 8 nM T89041 CC01FB 71454470 IC50 = 199 nM T89041 CG1CQ6 71454483 IC50 > 2500 nM T89041 C70TUP 71455138 IC50 > 10000 nM T89041 C70ARH 71456230 IC50 = 970 nM T89041 CFG4L5 71456934 IC50 > 10000 nM T89041 CX4U8V 71459926 IC50 = 1520 nM T89041 C0SU7M 71461598 IC50 = 1520 nM T89041 C7XIS4 71461624 IC50 = 430 nM T89041 C58SMB 71574941 IC50 = 260 nM T89041 CC09FQ 71574942 IC50 = 1346 nM T89041 CA2T5L 71574943 IC50 = 1886 nM T89041 C9MFZ7 71574944 IC50 = 610 nM T89041 CW73OE 71574945 IC50 > 5000 nM T89041 C70NHJ 71574946 IC50 = 1250 nM T89041 CLH83S 71574947 IC50 > 5000 nM T89041 CF71AB 71575030 IC50 > 5000 nM T89041 CCG1S5 71575031 IC50 > 5000 nM T89041 CH9WE7 71575032 IC50 > 5000 nM T89041 CO4ZQ7 71575033 IC50 = 493 nM T89041 CT86GV 71575034 IC50 = 1737 nM T89041 CKPV51 71621803 IC50 = 38000 nM T89041 C56LUJ 71716957 IC50 > 10000 nM T89041 CRP1G5 71733625 IC50 = 122000 nM T89041 C7V2LS 71733626 IC50 = 93700 nM T89041 C3J8DZ 71734667 IC50 = 130000 nM T89041 C48JAU 71735007 IC50 = 132000 nM T89041 CJE01S 71745100 IC50 > 10000 nM T89041 CX0WV5 71817943 IC50 = 64 nM T89041 CN1LU6 71817944 IC50 = 106 nM T89041 CGV4U3 71817945 IC50 = 523 nM T89041 CJ4L5G 71818086 IC50 = 147 nM T89041 COXA51 71818087 IC50 = 375 nM T89041 CP1A3M 71818088 IC50 = 454 nM T89041 CPJ42T 71818089 IC50 = 525 nM T89041 CAP03I 71818090 IC50 = 94 nM T89041 CO23PK 71818091 IC50 = 185 nM T89041 CL4X6A 71818092 IC50 = 11 nM T89041 CL8GK5 71818093 IC50 = 16 nM T89041 C4ZVG0 71818094 IC50 = 294 nM T89041 CH2GR0 71818232 IC50 = 1028 nM T89041 C0VGQ9 71818233 IC50 = 632 nM T89041 C5QRF2 71818234 IC50 = 1520 nM T89041 CCG7R3 72703685 IC50 = 480 nM T89041 CAU4Z0 72703889 IC50 = 2160 nM T89041 C56KEC 72703890 IC50 > 5000 nM T89041 CZB6E9 73345904 IC50 = 206 nM T89041 C5TD1Y 76335179 IC50 = 1800 nM T89041 C1YJW0 77846787 IC50 = 67 nM T89041 CV73PD 77846790 IC50 = 9 nM T89041 C0DIH7 77846872 IC50 = 15 nM T89041 COI25M 77846873 IC50 = 7 nM T89041 CJI8R0 77846875 IC50 = 8 nM T89041 CZK4J1 77846962 IC50 = 9 nM T89041 CEK89G 77846963 IC50 = 19 nM T89041 C5BA8Z 77846964 IC50 = 11 nM T89041 C4D6XJ 77847803 IC50 = 0.73 nM T89041 CF7O4Q 77847804 IC50 = 12 nM T89041 C3RHG9 85468997 IC50 = 480 nM T89041 CZH2O5 87178837 IC50 = 258000 nM T89041 CL30TR 89471870 IC50 > 10000 nM T89041 C3BUS8 89471889 IC50 > 10000 nM T89041 CI7HY8 89471890 IC50 = 5700 nM T89041 CX0M7B 89961716 IC50 = 84 nM T89041 CR5D6Y 89961785 IC50 > 10000 nM T89041 C89TEU 89968659 IC50 > 10000 nM T89041 CY5IC7 90252834 IC50 > 10000 nM T89041 C84NVA 90252850 IC50 > 10000 nM T89041 CBY46O 90252851 IC50 > 10000 nM T89041 CNVA50 90252852 IC50 > 10000 nM T89041 C89BFG 90333640 IC50 = 3.7 nM T89041 C0YK1U 90656806 IC50 = 310 nM T89041 CWE0X5 90656807 IC50 > 4000 nM T89041 CQS8C9 91664365 IC50 = 2 nM T89041 CLB2E7 91827654 IC50 > 10000 nM T89041 CN5ZQ2 117629963 IC50 > 15000 nM T89041 CJ9Z0S 118496546 IC50 > 10000 nM T89041 CJ54UQ 118618017 IC50 = 21 nM T89041 C7FT2M 118691578 IC50 = 22.8 nM T89041 CZD9X8 118691599 IC50 = 15.5 nM T89041 CDHI10 118733086 IC50 > 10000 nM T89041 C18PWB 118733087 IC50 > 10000 nM T89041 C8WJ2Y 118733088 IC50 > 10000 nM T89041 C31ZXP 118733089 IC50 > 10000 nM T89041 CHR84E 118733090 IC50 > 10000 nM T89041 CAQ72M 118733091 IC50 > 10000 nM T89041 CIV1Z5 118733092 IC50 > 10000 nM T89041 CU3Y9W 118733093 IC50 > 10000 nM T89041 CF49NU 118733094 IC50 > 10000 nM T89041 CK73VU 118733095 IC50 > 10000 nM T89041 CR1WU5 118733096 IC50 > 10000 nM T89041 CK7Y2L 118858329 IC50 = 230 nM T89041 CK09QT 118858331 IC50 = 12.4 nM T89041 C4CB3G 118867913 IC50 = 39000 nM T89041 CFND03 121481824 IC50 = 1 nM T89041 CO48UI 121481829 IC50 = 5 nM T89041 CM71FR 121481838 IC50 = 1 nM T89041 C48QHN 121481842 IC50 = 6.2 nM T89041 CMJB40 121481843 IC50 = 5 nM T89041 CMP69L 121481849 IC50 = 5 nM T89041 C02XEN 121481855 IC50 = 5 nM T89041 CRP3W8 121481856 IC50 = 5 nM T89041 CTE53N 121481871 IC50 = 17 nM T89041 C1GI5N 121481873 IC50 = 86 nM T89041 CYD80P 121481874 IC50 = 100 nM T89041 CX1FE7 121481875 IC50 = 39 nM T89041 C4XF6C 121481880 IC50 = 117 nM T89041 CBGY79 121481882 IC50 = 1200 nM T89041 CGA71F 121481885 IC50 = 42 nM T89041 C29AKG 121481886 IC50 = 5 nM T89041 C2NWZ7 121481888 IC50 = 180 nM T89041 C8IZ9B 121481891 IC50 = 2500 nM T89041 C8XO3C 121481900 IC50 = 58 nM T89041 C7SOX9 122439257 IC50 = 24 nM T89041 C15NCI 122439267 IC50 = 4.6 nM T89041 CP3K5Z 122439268 IC50 = 21 nM T89041 CX4T7L 122439274 IC50 = 5 nM T89041 CT9E7N 122439276 IC50 = 17 nM T89041 CSI91Y 122439277 IC50 = 18 nM T89041 C8EG3B 122439285 IC50 = 5 nM T89041 C80OLS 122462854 IC50 > 31622.78 nM T89041 C15JTL 122462980 IC50 > 31622.78 nM T89041 CUF8C5 126761305 IC50 = 7.83 nM T89041 C2ZFR8 127027572 IC50 > 10000 nM T89041 CV1BD6 127027573 IC50 > 10000 nM T89041 CQO36B 127028499 IC50 = 6600 nM T89041 CN42BR 127028817 IC50 > 10000 nM T89041 C49IME 127031799 IC50 = 4800 nM T89041 C6U0PW 127031978 IC50 = 5 nM T89041 C7EV5P 127031979 IC50 = 2 nM T89041 C6T5VG 127031980 IC50 = 5 nM T89041 CD1NK7 127031981 IC50 = 4 nM T89041 CX05HP 127032282 IC50 = 5 nM T89041 CP4WZ3 127033243 IC50 = 4 nM T89041 CNJW13 127034300 IC50 = 3 nM T89041 C2EO9D 129811602 IC50 > 20000 nM T89041 C74WZM 131748940 IC50 = 42 nM T89041 CH3V9Q 134139925 IC50 > 10000 nM T89041 C4DLP3 136029154 IC50 = 5900 nM T89041 CAV9U3 136219390 IC50 = 910 nM T89041 CC7LY3 136239517 IC50 = 550 nM T89041 C2V0IM 136244612 IC50 > 5000 nM T89041 CYIF59 136245971 IC50 > 5000 nM T89041 CG91VC 137633656 IC50 = 24.3 nM T89041 C4ALG0 137635843 IC50 = 20.1 nM T89041 C6Y8VD 137636260 IC50 = 45 nM T89041 CH2SR6 137636922 IC50 = 23.7 nM T89041 C6MJU7 137653906 IC50 = 45.4 nM T89041 CL45EH 137658689 IC50 = 29 nM T89041 C0ROV3 145961601 IC50 = 5 nM T89041 C63WHT 145961979 IC50 = 6 nM T89041 CVR84G 145962556 IC50 = 5 nM T89041 COPL56 145962564 IC50 = 5 nM T89041 CGP0Z7 145963339 IC50 = 34 nM T89041 CK71RV 145963932 IC50 > 31622.78 nM T89041 C74HIS 145965339 IC50 = 7.2 nM T89041 C9G2OD 145974857 IC50 = 16.5 nM T89041 CMW1H3 155544953 IC50 > 15000 nM T89041 D00DSE 49864196 IC50 = 386 nM T89041 D00IUN 25099145 IC50 = 953 nM T89041 D00YHD 46854449 IC50 = 783 nM T89041 D00ZME 9861000 IC50 = 4 nM T89041 D01REI 46901610 IC50 = 52 nM T89041 D01SZX 46867545 IC50 = 880 nM T89041 D02BXS 46901445 IC50 = 337 nM T89041 D03EDD 10593052 Ki = 41 nM T89041 D03EXD 49864181 IC50 = 248 nM T89041 D04CFP 46901927 IC50 = 760 nM T89041 D04ISG 11680597 IC50 = 27 nM T89041 D04SHY 42642719 IC50 = 195 nM T89041 D05LXA 44587266 IC50 = 310 nM T89041 D05PKT 46901928 IC50 = 2000 nM T89041 D06AKB 49864180 IC50 = 4040 nM T89041 D07CTI 10853186 IC50 = 130 nM T89041 D07IQG 10473365 IC50 = 42 nM T89041 D07VGT 46901929 IC50 = 438 nM T89041 D08FAB 11845485 IC50 = 3000 nM T89041 D08YCD 10354661 IC50 = 910 nM T89041 D09GEH 44587233 IC50 = 450 nM T89041 D09GJI 44586828 IC50 = 99 nM T89041 D09VQZ 46901616 IC50 = 598 nM T89041 D0B9XL 25099144 IC50 = 373 nM T89041 D0E0ZS 46901613 IC50 = 876 nM T89041 D0GJ7J 3760 Ki = 610 nM T89041 D0I1YH 46901446 IC50 = 97 nM T89041 D0J4VA 46854606 IC50 = 343 nM T89041 D0JE1I 9815923 IC50 > 19952.62 nM T89041 D0K5KG 6540050 IC50 = 1085 nM T89041 D0L6HY 20298212 IC50 = 2300 nM T89041 D0LJ9D 46901783 IC50 = 647 nM T89041 D0M8JE 13416469 IC50 = 780 nM T89041 D0MM7G 18976090 IC50 = 388 nM T89041 D0N1GH 11601068 IC50 = 686 nM T89041 D0N1PQ 11506923 IC50 = 667 nM T89041 D0N7CQ 42642718 IC50 = 152 nM T89041 D0P5CT 46901614 IC50 = 1790 nM T89041 D0Q0BK 46901611 IC50 = 186 nM T89041 D0Q1FX 42642717 IC50 = 164 nM T89041 D0Q1LG 44587267 IC50 = 300 nM T89041 D0RD3C 44587268 IC50 = 2100 nM T89041 D0RI7T 44586827 IC50 = 1400 nM T89041 D0SM4F 42642716 IC50 = 231 nM T89041 D0SP7S 5995 IC50 = 56 nM T89041 D0SU0Y 44587265 IC50 = 580 nM T89041 D0T1CH 46901440 IC50 = 1610 nM T89041 D0U5GF 18976091 IC50 = 282 nM T89041 D0U6JI 46854448 IC50 = 189 nM T89041 D0WN9P 46901444 IC50 = 226 nM T89041 D0X1DV 44587321 IC50 = 2000 nM T89041 D0Y5KX 46901443 IC50 = 408 nM T89041 D0Z3GX 46901784 IC50 = 577 nM T76522 CCYB38 206441 Ki = 22500 nM T76522 C4MRT6 16193817 IC50 > 10000 nM T76522 CKXV20 53434646 Ki = 125000 nM T76522 CM0CB3 71385905 Ki = 24000 nM T76522 CI5PJ9 71400937 Ki = 68100 nM T76522 CV7YP6 90655688 Ki = 105000 nM T76522 CKV18N 134146743 IC50 > 10000 nM T74307 D09KTS 24821094 IC50 = 0.23 nM T74307 D02TUL 118115473 IC50 = 19000 nM T74307 D08AOZ 86582336 IC50 = 23 nM T74307 D08UUL 46700756 IC50 = 4409 nM T74307 D0E3TC 44259 IC50 = 1.07 nM T74307 D0G5XV 135565884 IC50 = 1.13 nM T74307 D0H9FR 118295624 IC50 = 371 nM T74307 D0O6WV 24794418 IC50 > 500 nM T74307 D0YB3W 156414 IC50 = 29 nM T74307 D03BNU 59604787 IC50 > 10000 nM T74307 D09HEV 6539952 IC50 = 46 nM T74307 D0T3ME 156422 IC50 > 30000 nM T74307 CB7WK3 5938113 IC50 = 8800 nM T74307 CBOP58 11293798 Ki > 10000 nM T74307 C26BZX 11362471 Ki > 10000 nM T74307 CWXB93 11397177 Ki > 10000 nM T74307 C0APW4 11422034 IC50 = 10000 nM T74307 CTG83F 11539329 Ki > 1500 nM T74307 CMIL86 11590363 Ki > 1500 nM T74307 C9T6SC 11640926 Ki > 1500 nM T74307 CU0E8O 11690457 Ki > 10000 nM T74307 CB0AP2 11705863 Ki > 10000 nM T74307 CZY05V 11719421 IC50 = 1320 nM T74307 CP7AH3 11755812 IC50 = 50000 nM T74307 CFPW41 16007116 Ki > 1400 nM T74307 C9TU1O 16046126 IC50 > 1000 nM T74307 CQNP54 24764449 IC50 = 519 nM T74307 C3VRO9 44557921 IC50 > 10000 nM T74307 CY3HW5 46224684 IC50 = 8300 nM T74307 CLS29B 46872626 IC50 > 10000 nM T74307 C2O8RZ 46886323 IC50 = 320 nM T74307 C8NA4L 53384644 IC50 > 30000 nM T74307 CE1A9V 57394653 IC50 = 16 nM T74307 CI50KU 58167984 IC50 = 959 nM T74307 C1MR8Q 60097495 IC50 > 10000 nM T74307 CV63UL 67240318 IC50 > 10000 nM T74307 C7VJ6A 70647728 IC50 = 20 nM T74307 COU73Y 71226944 IC50 = 9 nM T74307 C40JOZ 71235465 IC50 = 78 nM T74307 CKT60L 71455860 Ki > 1400 nM T74307 CEV53L 71548006 IC50 = 32 nM T74307 C1SR5V 71576693 IC50 = 377 nM T74307 C4X1CP 71748056 IC50 = 366 nM T74307 CZM1K4 71765510 IC50 = 36 nM T74307 CKO8S6 71815907 IC50 = 339 nM T74307 CF6QG1 73602845 IC50 = 191 nM T74307 CDN83F 73707530 IC50 = 30.2 nM T74307 CCQN01 73775788 IC50 = 250 nM T74307 CHF08G 73775789 IC50 = 1130 nM T74307 COL37D 73775921 IC50 = 83.6 nM T74307 CVQW20 73775923 IC50 = 2060 nM T74307 C5U4AF 73776059 IC50 = 160 nM T74307 CXW54V 73776061 IC50 = 177 nM T74307 CD83FL 73776204 IC50 = 342 nM T74307 CG84BR 73776205 IC50 = 2090 nM T74307 C1P3DO 73776206 IC50 = 1950 nM T74307 CN5D1R 73776207 IC50 = 300 nM T74307 CO1C8Y 73776208 IC50 = 246 nM T74307 CGC46K 73776360 IC50 = 295 nM T74307 CN39OQ 78341183 IC50 = 22 nM T74307 C64SIO 92042864 IC50 = 157 nM T74307 CAKD54 102594000 IC50 > 10000 nM T74307 CJGT03 118346182 IC50 = 607 nM T74307 C02DGP 118346184 IC50 > 10000 nM T74307 CU6NE2 118346192 IC50 = 336 nM T74307 CW25VP 118346194 IC50 = 293 nM T74307 CQCX41 118737057 IC50 = 19 nM T74307 CDSV38 121316062 Ki = 190 nM T74307 C81IFQ 122163152 IC50 > 100000 nM T74307 C76IKM 122705261 IC50 > 100000 nM T74307 CG8DA9 127045861 IC50 > 100000 nM T74307 CC4ND8 127046862 IC50 > 100000 nM T74307 CIU72D 127264586 IC50 = 8.1 nM T74307 C6ROQ3 132546210 IC50 = 81 nM T74307 CXC69T 137321158 IC50 = 138 nM T74307 C3Z4AT 137321159 IC50 > 10000 nM T74307 CZOD53 137633880 IC50 = 53 nM T74307 C7BJY5 137636807 IC50 = 50 nM T74307 C4DRX1 137643187 IC50 = 3050 nM T74307 CO89DX 137649100 IC50 = 29 nM T74307 CINE03 137652514 IC50 = 280 nM T74307 C28QUP 137652864 IC50 = 76.4 nM T74307 CGW9I0 137656387 IC50 = 5260 nM T74307 C4OD9Q 145967187 IC50 = 0.2 nM T74307 CE31VG 145979714 IC50 > 10000 nM T74307 C9BX4U 145988956 IC50 > 10000 nM T74307 C2MD1Q 155513187 IC50 > 10000 nM T74307 CI23DH 155516489 IC50 = 198 nM T74307 C3NA2I 155519537 IC50 = 10 nM T74307 CY5MR2 155522337 Ki = 170 nM T74307 CL0US4 155530459 IC50 = 0.7 nM T74307 C78MZC 155536330 IC50 = 8 nM T74307 CZQM57 155554194 IC50 = 2713.75 nM T74307 D00ERW 44444843 Ki > 1453 nM T74307 D00HVA 11624601 Ki > 1500 nM T74307 D01RHR 71519693 IC50 = 2.7 nM T74307 D01VFR 4708 IC50 = 5470 nM T74307 D06BJG 71556703 IC50 = 4.2 nM T74307 D0GN5Z 5281295 IC50 = 2880 nM T74307 D0Q3NG 11715520 Ki > 1500 nM T74307 D0S7IE 11658882 Ki > 1500 nM T21865 D02AUB 9811353 IC50 = 70000 nM T21865 D0Z0AM 12004316 IC50 = 150000 nM T21865 C96KNY 643990 IC50 = 15000000 nM T21865 CM8YN2 11348172 IC50 = 413000 nM T21865 CTDH45 14498151 IC50 = 4000000 nM T21865 CZ13DK 14498163 IC50 = 1000000 nM T21865 CJE6Y0 16099896 IC50 = 1500000 nM T21865 CGK0T7 16099901 IC50 = 1500000 nM T21865 C8CUQ4 16099902 IC50 = 3000000 nM T21865 C8D0KF 16099905 IC50 = 450000 nM T21865 CM8CL1 16099913 IC50 = 400000 nM T21865 C3UK7A 16099914 IC50 = 250000 nM T21865 C3V2KY 16099916 IC50 = 700000 nM T21865 C31XCS 16099919 IC50 = 225000 nM T21865 C0U9ZL 16099921 IC50 = 1500000 nM T21865 C2FXW0 16099923 IC50 = 200000 nM T21865 C3W7YQ 16099925 IC50 = 2000000 nM T21865 CFY05L 16099926 IC50 = 375000 nM T21865 CO5SY7 16099929 IC50 = 625000 nM T21865 CR6W3S 16099936 IC50 = 1500000 nM T21865 C7E3WD 16099940 IC50 = 1000000 nM T21865 CI0GX1 16099943 IC50 = 1000000 nM T21865 C0L5FE 16099944 IC50 = 200000 nM T21865 C0T6OC 16099945 IC50 = 400000 nM T21865 CZS67I 16099962 IC50 = 2000000 nM T21865 C51NZE 16099968 IC50 = 75000 nM T21865 C2NH3G 16099971 IC50 = 125000 nM T21865 C0IBF1 16099978 IC50 = 300000 nM T21865 CK4IH9 16099980 IC50 = 240000 nM T21865 CZ2FH9 16099985 IC50 = 1000000 nM T21865 CUM26S 16100003 IC50 = 600000 nM T21865 C4ZVE0 16100004 IC50 = 550000 nM T21865 CUMK61 16100005 IC50 = 1600000 nM T21865 CDG5U9 16100006 IC50 = 625000 nM T21865 CN6EC7 16100010 IC50 = 300000 nM T21865 C4B7JV 16100012 IC50 = 525000 nM T21865 CBK6Z3 16100014 IC50 = 175000 nM T21865 C7VE4W 16100015 IC50 = 500000 nM T21865 C9BKC2 16100016 IC50 = 225000 nM T21865 C2FHQ1 16100024 IC50 = 250000 nM T21865 C80LWT 16100025 IC50 = 250000 nM T21865 CT7HP1 25103104 IC50 = 250000 nM T21865 CD9KM7 44287084 IC50 = 2500000 nM T21865 CUS84P 46915502 IC50 = 175000 nM T21865 C19MAV 135547550 IC50 = 3500000 nM T21865 D00YPH 10239 IC50 = 6000000 nM T22302 CL3K7I 5310497 IC50 = 1200 nM T22302 CGMN97 25067404 IC50 = 537 nM T22302 C9B6XI 70686297 IC50 = 385 nM T22302 C6TNB2 70690451 IC50 = 6900 nM T22302 C4GXP2 70690453 IC50 = 61 nM T22302 CRGC43 70694654 IC50 = 2900 nM T22302 C2QHP7 70694655 IC50 = 177 nM T22302 CORP75 70696691 IC50 = 570 nM T22302 CRY1E6 70696692 IC50 = 1057 nM T22302 C24ACH 70696693 IC50 = 640 nM T22302 D0M2PP 7211972 IC50 = 568 nM T18477 D01BYB 5957 IC50 = 861330 nM T18477 D0E7PQ 5311 IC50 > 1000 nM T18477 D01FYA 9549213 IC50 = 43 nM T18477 D02TTL 44156921 IC50 = 33 nM T18477 D05BYA 135539077 IC50 < 0.4 nM T18477 D05HWN 16736529 Ki = 1.7 nM T18477 D06YSP 11955716 IC50 = 13.6 nM T18477 D07MPL 44195571 IC50 = 38 nM T18477 D0F3NF 67501411 Ki = 34.7 nM T18477 D0I1QI 135564985 IC50 = 5 nM T18477 D0K5BP 46216556 IC50 = 13 nM T18477 D00OCB 984170 IC50 = 280 nM T18477 D00GOM 71453910 IC50 = 90 nM T18477 D09BVL 4552 IC50 = 3320 nM T18477 CG47UK 10241 IC50 > 1000 nM T18477 CTV6F8 107935 IC50 = 1630 nM T18477 CUM2L9 145989 IC50 > 1250000 nM T18477 CA23LP 448972 EC50 = 170 nM T18477 C07TEG 764764 IC50 = 4400 nM T18477 CXK79E 767613 IC50 = 4730 nM T18477 C4L6KE 2766290 IC50 = 9600 nM T18477 CB6OK2 5287464 IC50 = 15200 nM T18477 CI7MW0 9852185 IC50 = 21980 nM T18477 C7E9KA 10177135 EC50 = 160 nM T18477 CU9SK6 10183346 EC50 = 30 nM T18477 CB7D8O 11187955 EC50 = 310 nM T18477 CO3HN2 11189279 EC50 = 130 nM T18477 CYQP95 11198704 IC50 > 100000 nM T18477 CO3F6K 11221466 IC50 > 100000 nM T18477 CH4B2Z 11223683 IC50 > 200000 nM T18477 C9ZS0N 11247073 EC50 = 2000 nM T18477 CA45FP 11266813 IC50 = 28030 nM T18477 CBZS48 11302159 IC50 > 300000 nM T18477 C0L2WJ 11314518 IC50 = 23930 nM T18477 CDJX31 11326407 IC50 = 60400 nM T18477 C2ZCY3 11336657 IC50 > 300000 nM T18477 CIRH67 11349446 IC50 > 300000 nM T18477 CUO6Q7 11393625 IC50 > 100000 nM T18477 CXN76P 11406285 IC50 > 500000 nM T18477 CP3Z4O 11407267 IC50 > 100000 nM T18477 CZKO68 11407809 EC50 = 20 nM T18477 CIG8V3 11415875 EC50 = 98 nM T18477 CP90LC 11427896 IC50 > 100000 nM T18477 CR9IQ7 11450570 IC50 > 300000 nM T18477 C8VZQ6 11463506 IC50 > 100000 nM T18477 CI53RD 11473241 IC50 > 100000 nM T18477 CQL4M5 11475629 EC50 = 4300 nM T18477 C6S3TY 11488262 EC50 = 470 nM T18477 C9IY1M 11517212 Ki = 0.2 nM T18477 CKSG91 11751343 EC50 = 90 nM T18477 C79VTC 11773074 IC50 > 50000 nM T18477 CPB49N 11855206 Ki = 235 nM T18477 CR1X7L 11950337 IC50 = 0.7 nM T18477 CAGU13 11950510 EC50 = 9 nM T18477 C8WAX9 11957092 Ki = 700 nM T18477 CE8M7K 12318923 IC50 = 31000 nM T18477 C8M6SA 12331235 IC50 = 13300 nM T18477 C82YHV 12331237 IC50 = 14900 nM T18477 CG07VM 12331240 IC50 = 49600 nM T18477 C4G8MJ 12571204 IC50 = 750 nM T18477 C9C4WH 15856427 IC50 = 24000 nM T18477 C7RCT2 15856428 IC50 = 16000 nM T18477 CDFK08 16061445 IC50 = 54 nM T18477 CI14ZN 16225982 IC50 = 19 nM T18477 C6JY5F 16226184 IC50 = 10 nM T18477 CTRL63 16667105 EC50 = 250 nM T18477 C1EXG6 16727212 IC50 = 220 nM T18477 C3BXP9 17545684 IC50 = 13300 nM T18477 CPYW42 21179452 IC50 = 42200 nM T18477 CRA65J 21846414 IC50 = 6900 nM T18477 CAS5G3 23958192 IC50 = 16.82 nM T18477 C7RTS1 24768274 IC50 > 20000 nM T18477 C7P4RL 24768277 IC50 > 20000 nM T18477 C1T4WH 25003030 Ki = 11 nM T18477 COBM26 25073055 IC50 = 28 nM T18477 C8F1MA 44323467 IC50 = 33000 nM T18477 CM5XT0 44376308 EC50 = 3600 nM T18477 C8WJ9S 44376565 EC50 = 1400 nM T18477 CAKW20 44376753 EC50 = 3500 nM T18477 CSHJ14 44383813 EC50 > 50000 nM T18477 C45XQM 44400015 EC50 = 330 nM T18477 C0L5XP 44400119 EC50 = 2800 nM T18477 C2UWT8 45162180 IC50 = 308500 nM T18477 C3BJ9O 45788206 Ki = 8300 nM T18477 CS6J7Q 46861552 Ki = 1200 nM T18477 CSD39K 46912795 IC50 = 94 nM T18477 CRIB76 46913258 IC50 = 365 nM T18477 C8U9LT 46919029 IC50 = 490 nM T18477 C15CFW 46919030 IC50 = 510 nM T18477 CUP92O 49842657 IC50 = 585 nM T18477 C54HZQ 49863672 IC50 = 1400 nM T18477 CE4AN1 49863673 IC50 = 650 nM T18477 C0U8MW 49863674 IC50 = 5100 nM T18477 C6T9HE 49863675 IC50 = 790 nM T18477 C19VJH 49863676 IC50 = 3400 nM T18477 CX74OK 49863677 IC50 = 1100 nM T18477 C0Q8ZV 49863678 IC50 = 3100 nM T18477 C21JZL 49870746 IC50 = 9524 nM T18477 CBA6D2 49871894 IC50 = 470 nM T18477 CR0U5H 49871895 IC50 = 58 nM T18477 C2ERZ4 49871985 IC50 = 183 nM T18477 CMA10L 49871988 IC50 = 750 nM T18477 C7GRS3 50925477 EC50 = 60 nM T18477 C2OVL4 51049656 Ki = 130 nM T18477 C4MZ7N 52916002 IC50 = 15530 nM T18477 CK98TP 52918129 IC50 = 90 nM T18477 CB1JE7 52918144 IC50 = 110 nM T18477 CHZP24 53236116 Ki = 190 nM T18477 C3MA7Q 53236117 Ki = 120 nM T18477 C3RCQ9 53236118 Ki = 16 nM T18477 CLPO19 53236119 Ki = 250 nM T18477 C2BYJ6 53236120 Ki = 7 nM T18477 C7OSD2 53236121 Ki = 35 nM T18477 C8G5TM 53236346 Ki = 20 nM T18477 CL60TN 53236347 Ki = 13 nM T18477 CU1BE9 53236348 Ki = 12 nM T18477 CFL65I 53236349 Ki = 9 nM T18477 CV7BK2 53236350 Ki = 6 nM T18477 CH8LV9 53236351 Ki = 9 nM T18477 CQM95X 53236589 Ki = 7 nM T18477 CFI32H 53239287 Ki = 50 nM T18477 C35TQX 53239288 Ki = 26 nM T18477 CJ68VG 53239289 Ki = 38 nM T18477 CGMZ76 53239290 Ki = 21 nM T18477 CG26RE 53239291 Ki = 18 nM T18477 C1VJ0T 53239502 Ki = 7 nM T18477 C80QGZ 53239503 Ki = 110 nM T18477 CYC7B4 53239504 Ki = 7 nM T18477 C4S8QK 53239505 Ki = 27 nM T18477 CTJB43 53239506 Ki = 40 nM T18477 C13XHA 53239507 Ki = 300 nM T18477 CKNJ47 53245660 IC50 = 83 nM T18477 CW9IQ0 53248730 IC50 = 82 nM T18477 CVHW83 53259029 IC50 = 110 nM T18477 C1KYR9 53326941 IC50 = 96 nM T18477 CI0R4B 54580554 IC50 = 96 nM T18477 CRV6M8 54580555 IC50 = 126 nM T18477 CYC3K8 54580556 IC50 = 3324 nM T18477 CYC3V7 54580557 IC50 = 153 nM T18477 C34EOA 54580558 IC50 = 301 nM T18477 CRF0G6 54581044 IC50 = 830 nM T18477 CA3CX5 54581045 IC50 = 320 nM T18477 CHFD41 54581046 IC50 = 150 nM T18477 C4EH1F 54581551 IC50 = 201 nM T18477 CYAI91 54581552 IC50 = 634 nM T18477 CA73VM 54581553 IC50 = 496 nM T18477 CIHT85 54582089 IC50 > 5000 nM T18477 CZG19I 54582090 IC50 = 1240 nM T18477 CBI7N9 54582551 IC50 > 5000 nM T18477 C15SZU 54582552 IC50 = 188 nM T18477 CONG87 54582553 IC50 = 982 nM T18477 CF87RH 54583025 IC50 = 210 nM T18477 CEOZ15 54583522 IC50 = 96 nM T18477 CW2AF0 54584037 IC50 = 400 nM T18477 CQ65AR 54584038 IC50 = 570 nM T18477 C96JOM 54584500 IC50 = 883 nM T18477 CJV94T 54584501 IC50 = 78 nM T18477 C1T5NF 54584983 IC50 = 12440 nM T18477 CNJO03 54584984 IC50 > 5000 nM T18477 C96JXE 54585939 IC50 = 430 nM T18477 CSC0H3 54586414 IC50 = 61 nM T18477 C7HD0U 54586415 IC50 = 170 nM T18477 CFI5J2 54586912 IC50 = 290 nM T18477 C7G6IP 54586913 IC50 = 140 nM T18477 CZK7F1 54586914 IC50 = 920 nM T18477 CZ54WE 54586915 IC50 = 360 nM T18477 CD06RB 54587434 IC50 = 106 nM T18477 CR1I6J 54587584 IC50 = 145 nM T18477 CM01DQ 54764333 IC50 = 5600 nM T18477 C2QK8U 56659496 IC50 = 24800 nM T18477 CA9T4B 56659497 IC50 = 25200 nM T18477 CC8AZ2 56659584 IC50 = 80 nM T18477 C6QSI8 56659760 IC50 = 84 nM T18477 C71GNP 56659879 IC50 > 200000 nM T18477 CWKH97 56659880 IC50 > 200000 nM T18477 C01XAG 56662951 IC50 = 15400 nM T18477 COEU61 56662986 IC50 = 34900 nM T18477 C1RPG4 56662987 IC50 = 200000 nM T18477 CL8J5E 56663234 IC50 = 82 nM T18477 CS0OL3 56663235 IC50 = 88 nM T18477 CK81DA 56663236 IC50 = 74 nM T18477 CASK95 56663304 IC50 = 116 nM T18477 CF3DM2 56663339 IC50 > 200000 nM T18477 C28OQJ 56666428 IC50 = 72 nM T18477 CW51JK 56666664 IC50 = 116 nM T18477 C5XGS1 56666665 IC50 = 142 nM T18477 CFI5R6 56666666 IC50 = 66 nM T18477 C3D4TK 56666731 IC50 = 83 nM T18477 CYQE09 56666732 IC50 = 65 nM T18477 CEU56I 56666733 IC50 = 68 nM T18477 CA3HM7 56666734 IC50 = 228 nM T18477 CCR76H 56670085 IC50 = 64 nM T18477 C6EFP7 56670086 IC50 = 85 nM T18477 C0ABN1 56670087 IC50 = 77 nM T18477 CX92TP 56670157 IC50 = 83 nM T18477 CU6CS9 56670202 IC50 > 200000 nM T18477 C24YWF 56670203 IC50 > 200000 nM T18477 CXUI30 56673328 IC50 = 47 nM T18477 CD65HO 56673605 IC50 = 58 nM T18477 CFOE91 56673671 IC50 = 60 nM T18477 C3KZM9 56673672 IC50 = 91 nM T18477 CEN4H5 56676988 IC50 = 70 nM T18477 CI0Y5Z 56677032 IC50 > 200000 nM T18477 C10YJZ 56679993 IC50 = 33 nM T18477 C4AOI1 56679994 IC50 = 27 nM T18477 C1BPY4 56680021 IC50 = 127000 nM T18477 CW4JM5 56680236 IC50 = 81 nM T18477 CG34TX 56680322 IC50 = 183 nM T18477 CG51ZV 56681935 IC50 = 570 nM T18477 COL34U 56683638 IC50 = 131 nM T18477 CPMG31 56683692 IC50 > 200000 nM T18477 C73AOX 57404605 IC50 = 23 nM T18477 CM89YZ 57404775 IC50 = 27 nM T18477 CTQ1N2 57404776 IC50 = 95 nM T18477 CT65MO 57404777 IC50 = 270 nM T18477 CN0B1D 57405452 IC50 = 17 nM T18477 CT87RM 57406669 IC50 = 37 nM T18477 CD5C0Y 57406670 IC50 = 27 nM T18477 CO4W8R 57406671 IC50 = 36 nM T18477 C0RKH7 57406855 IC50 < 5 nM T18477 C8N1XS 57406856 IC50 = 23 nM T18477 CW1LY5 57406857 IC50 < 5 nM T18477 CI4C2X 57406859 IC50 = 21 nM T18477 CEH2P1 57406860 IC50 = 25 nM T18477 C3WPF1 57407047 IC50 < 5 nM T18477 CWH2N3 57407048 IC50 < 5 nM T18477 C3UN0J 57407049 IC50 < 5 nM T18477 C6I1SA 57407050 IC50 = 14.8 nM T18477 CA6Q1L 57407243 IC50 = 6.8 nM T18477 CP8AF0 57407244 IC50 = 15 nM T18477 CIJE49 57407246 IC50 = 32 nM T18477 CX9H1U 57407247 IC50 = 13 nM T18477 CTXS05 57407248 IC50 < 5 nM T18477 CH3OR8 57424824 IC50 = 300 nM T18477 CD56FL 57424831 IC50 = 56 nM T18477 C1L5UN 57424851 IC50 = 24 nM T18477 C70OWD 57424917 IC50 = 16 nM T18477 CI2WK1 57424929 IC50 > 10000 nM T18477 C3WLV1 57450675 IC50 = 37 nM T18477 CA4Y5Q 57450676 IC50 = 12 nM T18477 CU62HN 57450694 IC50 = 9800 nM T18477 C4G9FJ 57462510 IC50 = 27 nM T18477 CZVS05 57462516 IC50 = 140 nM T18477 CY87RC 57713841 IC50 = 3.9 nM T18477 C2FY4H 57748464 IC50 = 641 nM T18477 CSA3O2 57748552 IC50 = 479 nM T18477 C3HW6F 58762794 IC50 = 97 nM T18477 CZ7XQ5 60165612 Ki = 1800 nM T18477 CAU06M 66576834 IC50 = 100 nM T18477 C60LFE 66612138 IC50 = 27340 nM T18477 CV8B0R 67495834 Ki = 3 nM T18477 C2S9CE 67500027 IC50 = 73 nM T18477 C7IXO4 67500163 IC50 = 131 nM T18477 CZ2L9M 67500276 IC50 = 789 nM T18477 C0A6OX 67500939 IC50 = 52 nM T18477 C6VE3A 67500997 IC50 = 132 nM T18477 CD75KX 67501021 IC50 = 98 nM T18477 CPZA60 67501051 IC50 > 10000 nM T18477 CAX0I7 67501291 IC50 = 166 nM T18477 C32UVO 67502140 IC50 = 1168 nM T18477 CN26RP 67502287 IC50 = 1620 nM T18477 CX7G8L 67502777 IC50 = 72 nM T18477 C80ODY 67932020 Ki = 1380 nM T18477 C9TN8Q 67984974 IC50 = 35 nM T18477 CW4EM0 67985170 IC50 = 23 nM T18477 C4VT3I 67985199 IC50 = 30 nM T18477 C7WH6F 67985284 IC50 = 10 nM T18477 CQI6F7 67985727 IC50 < 5 nM T18477 CNC49F 71463004 IC50 = 1 nM T18477 CIG6P3 71660550 IC50 > 500000 nM T18477 C79AGJ 71660551 IC50 = 27300 nM T18477 CELO13 72376512 IC50 = 47000 nM T18477 CR3K1V 72547522 Ki = 2800 nM T18477 C9CW5M 73437615 Ki = 20 nM T18477 CUD54E 73437616 Ki = 5 nM T18477 CAW01J 74027120 IC50 = 22400 nM T18477 CUOW40 74222622 IC50 = 890 nM T18477 CRA86Z 76311786 IC50 = 48500 nM T18477 CJ2PU1 76315352 IC50 = 7600 nM T18477 CS97VJ 76315353 IC50 = 13200 nM T18477 CH0AP5 76319024 IC50 = 7400 nM T18477 CU3G6Q 76322418 IC50 = 12700 nM T18477 C68TOV 76322671 IC50 = 17300 nM T18477 C9BCH0 76322676 IC50 = 12700 nM T18477 CS0PB2 76324772 Ki = 125 nM T18477 CPX91U 76329863 IC50 = 26600 nM T18477 C2I4XM 76333294 IC50 = 12000 nM T18477 C49ZCD 76333509 IC50 = 16400 nM T18477 C6LV9H 76899944 IC50 = 410 nM T18477 CYZN80 76899957 IC50 = 470 nM T18477 C6WE9Y 77107768 IC50 = 1840 nM T18477 CAGX72 78106056 IC50 = 14330 nM T18477 C2N3CM 78106057 IC50 = 35240 nM T18477 CV2C8Q 78106150 IC50 = 8520 nM T18477 C47XUW 86280454 Ki > 100000 nM T18477 CT80DA 86294728 IC50 = 38 nM T18477 C2N7AP 86294734 IC50 = 70 nM T18477 C1ZKP7 86294735 IC50 = 38 nM T18477 CK98UO 86294736 IC50 = 21 nM T18477 C2MC0R 86294737 IC50 = 39 nM T18477 C40LNZ 86294738 IC50 = 190 nM T18477 CC3I7E 86302592 IC50 = 110 nM T18477 CVL4I0 86302593 IC50 = 29 nM T18477 C06YBD 86302594 IC50 = 33 nM T18477 CJ3Q4H 90654630 Ki = 6 nM T18477 CG8S1L 90654631 Ki = 3 nM T18477 CDIY85 90654632 Ki = 34 nM T18477 CV9YA4 90654633 Ki = 56 nM T18477 CRH14E 90654634 Ki = 180 nM T18477 C26WSJ 90654635 Ki = 94 nM T18477 CXLQ38 90654636 Ki = 14 nM T18477 C9F5UB 90654637 Ki = 10 nM T18477 CZ2MP4 90654638 Ki = 20 nM T18477 C17RWB 90654639 Ki = 40 nM T18477 C7X8WK 90654640 Ki = 32 nM T18477 CJ2ZM3 90654641 Ki = 42 nM T18477 C21FPZ 90654642 Ki = 14 nM T18477 C9ZTU1 90654643 Ki = 17 nM T18477 CTB60Y 90654644 Ki = 62 nM T18477 C81JGB 90654645 Ki = 28 nM T18477 CKM2W0 90654646 Ki = 22 nM T18477 CS8U1X 90654647 Ki = 46 nM T18477 CUE4I6 90654648 Ki = 28 nM T18477 CM5JP8 90654649 Ki = 28 nM T18477 CH8FD0 90654650 Ki = 25 nM T18477 C5DP2C 90654651 Ki = 22 nM T18477 CU87TN 90654652 Ki = 37 nM T18477 C4PJ1V 90654653 Ki > 10000 nM T18477 C2TYR0 90654654 Ki = 680 nM T18477 C6SI7L 90654655 Ki > 10000 nM T18477 CG2JK7 90654656 Ki = 390 nM T18477 CBWT05 90654657 Ki = 42 nM T18477 C6SK1Z 90654658 Ki = 36 nM T18477 C2TLY1 90654659 Ki > 10000 nM T18477 C3R1DJ 90654660 Ki = 1900 nM T18477 CT1QI5 90654661 Ki > 10000 nM T18477 CU8Q1V 90654662 Ki > 10000 nM T18477 CS42OM 90654663 Ki = 2500 nM T18477 C7M8TA 90654664 Ki = 3200 nM T18477 C1H5WC 90654665 Ki = 690 nM T18477 C9NO7L 90655134 IC50 = 34 nM T18477 C4SR1G 90655135 IC50 = 54 nM T18477 C18XMN 90655136 IC50 = 68 nM T18477 C82SQK 90655137 IC50 = 100 nM T18477 CEU4P7 90655138 IC50 = 160 nM T18477 C80KYO 90655139 IC50 = 1200 nM T18477 C29HUJ 90655140 IC50 = 1400 nM T18477 C6C7ST 90655141 IC50 = 3900 nM T18477 CGA47I 90655142 IC50 > 100000 nM T18477 C68KOR 90655143 IC50 > 100000 nM T18477 C3XL9Q 90655144 IC50 > 100000 nM T18477 CSR56C 90655296 IC50 = 31 nM T18477 C5WZ0F 90655297 IC50 = 12 nM T18477 C9HF1A 90655298 IC50 = 33 nM T18477 CW1UR6 90655299 IC50 = 181 nM T18477 CQ0JR2 90655300 IC50 > 1000 nM T18477 C76DSY 90655301 IC50 = 320 nM T18477 CZV1W0 90655302 IC50 = 295 nM T18477 C0UP3C 90656478 IC50 = 630 nM T18477 CQU83E 90656479 IC50 = 130 nM T18477 CW7L0S 90656480 IC50 = 330 nM T18477 CJY51L 90656481 IC50 = 130 nM T18477 CZ1I8E 90656482 IC50 = 250 nM T18477 CUD9J1 90656483 IC50 = 1500 nM T18477 CK94EB 90656484 IC50 = 130 nM T18477 C8R9JB 90656485 IC50 = 620 nM T18477 CWC3J9 90656486 IC50 = 78 nM T18477 CGL40M 90656487 IC50 = 71 nM T18477 CD6Z7W 90657117 Ki = 86 nM T18477 CI90DU 117736689 IC50 = 55 nM T18477 CVDP67 117736692 IC50 = 48 nM T18477 C60TAF 117736697 IC50 = 96 nM T18477 CX31TW 117736731 IC50 = 54 nM T18477 C2W9GO 117736733 IC50 = 91 nM T18477 CUVD12 117889758 IC50 > 25000 nM T18477 CUTV54 117889766 IC50 > 50000 nM T18477 CIBF07 117889785 IC50 > 100000 nM T18477 CW8J2A 117889863 IC50 > 100000 nM T18477 CP0VL5 117889908 IC50 = 24900 nM T18477 C0GZD8 117889984 IC50 > 100000 nM T18477 CGM51T 117890044 IC50 > 50000 nM T18477 C37QWO 117890084 IC50 > 50000 nM T18477 C1APC8 117890111 IC50 = 15970 nM T18477 CZ4EN5 117890133 IC50 > 50000 nM T18477 CO2R1E 117890146 IC50 > 100000 nM T18477 CE69YR 117890174 IC50 > 100000 nM T18477 C3C6KX 117890187 IC50 = 8300 nM T18477 CX6V7Q 117890195 IC50 > 50000 nM T18477 C4MQ8T 117890212 IC50 > 50000 nM T18477 CG53QV 117890216 IC50 = 20300 nM T18477 CZ45SB 117890250 IC50 > 100000 nM T18477 CLH49C 117890268 IC50 > 50000 nM T18477 CLHP30 117890308 IC50 > 100000 nM T18477 CQK30X 117890321 IC50 > 50000 nM T18477 CPWS97 117890346 IC50 > 50000 nM T18477 C1HK7L 117890351 IC50 > 50000 nM T18477 CO25TC 117890352 IC50 > 100000 nM T18477 CA15DJ 117890354 IC50 > 50000 nM T18477 CTV53C 117890368 IC50 = 1960 nM T18477 CQCT02 117890387 IC50 > 50000 nM T18477 CQ20HF 117890473 IC50 > 50000 nM T18477 C3R9DT 117890494 IC50 > 100000 nM T18477 CRYX09 117890515 IC50 > 50000 nM T18477 CK15CW 117967655 Ki = 9150 nM T18477 CQ4FL0 117968039 Ki = 3480 nM T18477 CYG8C4 117970892 Ki = 1980 nM T18477 CZ2AI8 117972517 Ki = 1020 nM T18477 CFI2P0 117972524 Ki = 6550 nM T18477 C5TFJ0 117972658 Ki = 3210 nM T18477 CN08WT 118712080 IC50 = 1040 nM T18477 CVK84L 118712081 IC50 = 430 nM T18477 C9A2OU 118719939 IC50 = 970 nM T18477 C6BGJ8 118720311 IC50 = 290 nM T18477 CXB34W 118724182 IC50 = 16 nM T18477 CG0R3L 118728263 Ki = 150 nM T18477 C3A8PL 118728264 Ki = 64 nM T18477 CKXV89 118728265 Ki = 213 nM T18477 COV7S8 118728266 Ki = 110 nM T18477 C3F7KR 118728267 Ki = 33 nM T18477 CX1DZ2 118728268 Ki = 54 nM T18477 C5TP4Q 118728269 Ki = 86 nM T18477 CX6U2K 118728270 Ki = 190 nM T18477 CRY17Z 118728271 Ki = 41 nM T18477 CTC60M 118728272 Ki = 50 nM T18477 CJT25I 118728273 Ki = 370 nM T18477 C9AT5X 118729959 Ki = 115 nM T18477 CDZ98W 118729960 Ki = 60 nM T18477 C5C8GB 118729961 Ki = 111 nM T18477 CKE49U 118737375 IC50 > 50000 nM T18477 C84YNW 118737376 IC50 > 50000 nM T18477 CKB9N5 118737377 IC50 > 50000 nM T18477 C1ZSK4 118737378 IC50 > 50000 nM T18477 CO6N4H 118796335 IC50 = 5 nM T18477 CBK28I 124081275 IC50 > 100000 nM T18477 CQ82GU 124201644 Ki = 10600 nM T18477 CCD60J 126962311 IC50 > 1000 nM T18477 CAQL68 126962384 IC50 > 1000 nM T18477 C59DWI 126962385 IC50 > 1000 nM T18477 CBXH95 127024111 Ki > 50000 nM T18477 CS1ZO6 127024161 Ki = 2510 nM T18477 CHQ12D 127024491 Ki > 50000 nM T18477 CBS1R8 127024554 Ki = 1780 nM T18477 CR6A9C 127024644 Ki > 50000 nM T18477 CGO8S5 129900226 IC50 = 698 nM T18477 CQ4S3Z 130277442 IC50 = 362 nM T18477 CX0QS8 130277744 IC50 = 611.5 nM T18477 C15ECZ 130277802 IC50 = 6.5 nM T18477 CW0D2F 131704417 IC50 = 36 nM T18477 CI47VP 131704472 IC50 = 39200 nM T18477 C0IQ4V 132601722 IC50 = 3680 nM T18477 CE3X8V 132992912 Ki > 13000 nM T18477 C4FPW8 132992920 Ki = 840 nM T18477 CUF85A 134132715 IC50 = 51 nM T18477 C1P5TE 134135478 IC50 = 94 nM T18477 CDC41Q 134138735 IC50 = 58 nM T18477 CH8G2J 134139194 IC50 = 79 nM T18477 CAB93T 134139543 IC50 = 750 nM T18477 C1PZ6L 134140295 IC50 = 480.8 nM T18477 CRDK20 134142142 IC50 = 183.3 nM T18477 CB7A0W 134145703 IC50 = 48 nM T18477 C0C4JZ 134147224 IC50 = 135.9 nM T18477 CC43OQ 134149366 IC50 = 50.3 nM T18477 CZEO76 134150482 IC50 = 8700 nM T18477 CZ68GA 134154630 IC50 > 1000 nM T18477 CT87WB 134156050 IC50 = 650 nM T18477 C0ZVI9 134157119 IC50 > 1000 nM T18477 CA0MT1 134480068 IC50 = 8932 nM T18477 CBRN70 135400938 IC50 = 60 nM T18477 CWHX62 135423284 IC50 = 62 nM T18477 CHZD50 135425202 IC50 = 210 nM T18477 CA1MC6 135433906 IC50 = 190 nM T18477 CS8JP3 135481178 IC50 = 150 nM T18477 C9NH7L 135499841 IC50 = 53 nM T18477 CVZ37K 135507483 IC50 = 120 nM T18477 C9EIC5 135507502 IC50 = 70 nM T18477 CK7PL9 135519368 IC50 = 510 nM T18477 C23HTX 135524913 IC50 = 39 nM T18477 CEK31P 135566415 IC50 = 30 nM T18477 CVJ05Z 135566858 IC50 = 70 nM T18477 CDIR12 135566860 IC50 = 27 nM T18477 CHE38I 135566861 IC50 = 23 nM T18477 C39USJ 135567370 IC50 = 37 nM T18477 CW54FS 135567371 IC50 = 38 nM T18477 C0QF7Z 135567372 IC50 = 42 nM T18477 CL59TN 135567373 IC50 = 44 nM T18477 C9KGT3 135567374 IC50 = 53 nM T18477 C1UEK8 135581701 IC50 = 40 nM T18477 CN97EY 135581702 IC50 = 800 nM T18477 CI85ZN 135981701 IC50 = 14500 nM T18477 C5J3KX 135981702 IC50 = 22100 nM T18477 CYV84F 136000662 Ki = 1400 nM T18477 C3ZBM8 136110909 IC50 = 66 nM T18477 CG06VA 136110910 IC50 = 121 nM T18477 C63FBA 136110911 IC50 = 57 nM T18477 CX27KJ 136110912 IC50 = 69 nM T18477 C5GD7K 136110913 IC50 = 295 nM T18477 CHQ05G 136110914 IC50 = 40 nM T18477 C3Y8LO 136110915 IC50 = 1660 nM T18477 CU8T5Q 136110916 IC50 = 546 nM T18477 CG2PO0 136110917 IC50 = 108 nM T18477 CUQ0B5 136110919 IC50 = 471 nM T18477 C1Y5HJ 136110920 IC50 = 307 nM T18477 CFPA47 136110921 IC50 = 99 nM T18477 CU6F1X 136110922 IC50 = 183 nM T18477 C8N1QK 136167232 Ki = 32 nM T18477 C2SRX9 136198647 IC50 > 100000 nM T18477 CEX34H 136198648 IC50 > 100000 nM T18477 CN0XY9 136198649 IC50 > 100000 nM T18477 CP79HX 136198650 IC50 > 100000 nM T18477 CR3LD9 136198651 IC50 > 100000 nM T18477 CN83ZX 136198652 IC50 > 100000 nM T18477 CEWC75 136198653 IC50 > 100000 nM T18477 C2NOH9 136236968 IC50 > 250000 nM T18477 CNM6L0 136266479 IC50 = 17 nM T18477 C0D6OT 136266481 IC50 = 35 nM T18477 C5SZ6I 136266482 IC50 = 46 nM T18477 CV7YO5 136266483 IC50 = 29 nM T18477 C8K5DR 136266484 IC50 = 57 nM T18477 C37HLR 136266485 IC50 = 36 nM T18477 C6XHU2 136266487 IC50 = 35 nM T18477 C4FLS0 136266488 IC50 = 27 nM T18477 C8G1CX 136266497 IC50 = 58 nM T18477 C0H9TJ 136266498 IC50 = 55 nM T18477 CDC53A 136266499 IC50 = 140 nM T18477 CKP7A9 136266500 IC50 = 30 nM T18477 CAPE16 136266501 IC50 = 44 nM T18477 C5XW9N 136266513 IC50 = 53 nM T18477 C7PCL8 136266514 IC50 = 44 nM T18477 C9NOM4 136266515 IC50 = 60 nM T18477 CO1U4Q 136266516 IC50 = 43 nM T18477 CL8MY2 136266517 IC50 = 35 nM T18477 C5LB9C 136266518 IC50 = 88 nM T18477 C5I3SJ 136266519 IC50 = 180 nM T18477 C05RDT 136266522 IC50 = 59 nM T18477 CJ3FE1 136266530 IC50 = 140 nM T18477 C1RP5H 136266531 IC50 = 42 nM T18477 CD9O8U 136266533 IC50 = 300 nM T18477 C2N5HF 136266558 IC50 = 70 nM T18477 C01ZXH 136266559 IC50 = 21 nM T18477 CTCO28 136934953 IC50 > 100000 nM T18477 CMZ90X 136934954 IC50 > 100000 nM T18477 CW40ER 136934955 IC50 > 100000 nM T18477 CKS79P 136934956 IC50 > 100000 nM T18477 CA4OC9 136934957 IC50 > 500000 nM T18477 CI8FR0 136934958 IC50 > 250000 nM T18477 C5VIG4 136934959 IC50 > 100000 nM T18477 C2YZ6E 136934960 IC50 > 100000 nM T18477 C6B4DY 136934961 IC50 > 100000 nM T18477 C01EUC 137069409 IC50 = 127 nM T18477 C0KZD3 137069410 IC50 = 50 nM T18477 COZ20T 137069411 IC50 = 78 nM T18477 C81TKF 137069412 IC50 = 120 nM T18477 C9PDL7 137069413 IC50 = 1660 nM T18477 CKH8P9 137069414 IC50 = 546 nM T18477 CB3P2W 137069415 IC50 = 66 nM T18477 CE35LW 137069416 IC50 = 207 nM T18477 CEL0H2 137069417 IC50 = 45 nM T18477 C7PGC2 137069418 IC50 = 144 nM T18477 CGWX25 137069419 IC50 = 114 nM T18477 CZX7K1 137069420 IC50 = 28 nM T18477 CFOU34 137069421 IC50 = 91 nM T18477 C18RKL 137069422 IC50 = 48 nM T18477 CG05CN 137069423 IC50 = 66 nM T18477 C2GB4N 137069424 IC50 = 33 nM T18477 CYF42G 137069425 IC50 = 54 nM T18477 CTG86A 137069426 IC50 = 152 nM T18477 C4ZM0V 137069427 IC50 = 125 nM T18477 CQEZ48 137069428 IC50 = 347 nM T18477 CZ8IH9 137069429 IC50 = 45 nM T18477 CTI86X 137069430 IC50 = 108 nM T18477 C5GKE7 137069431 IC50 = 66 nM T18477 CRL7Z3 137287446 IC50 > 1000 nM T18477 C8ZP0L 137440573 IC50 > 1000 nM T18477 C8V9ER 137440575 IC50 = 5.3 nM T18477 CD5H0E 137440576 IC50 = 413 nM T18477 CR60OH 137440582 IC50 = 995 nM T18477 CK0S4Q 137440583 IC50 = 429 nM T18477 CZW8E2 137440584 IC50 = 11.4 nM T18477 C9J2MH 137440585 IC50 = 830 nM T18477 C3O9BW 137440587 IC50 = 585 nM T18477 CRS03O 137440588 IC50 = 496 nM T18477 CAT74Q 137440592 IC50 = 558 nM T18477 C5QYW2 137440596 IC50 = 454 nM T18477 CZ54WU 137440598 IC50 > 1000 nM T18477 C3IT5C 137440602 IC50 = 528 nM T18477 CN26IS 137440610 IC50 = 135 nM T18477 CXF50C 137632543 IC50 > 1000 nM T18477 C9BX6Y 137635266 IC50 = 374 nM T18477 C39AGH 137635456 IC50 = 852 nM T18477 CC1DT5 137636870 IC50 = 307 nM T18477 CQ02SA 137637101 IC50 = 528 nM T18477 CKEW37 137638689 IC50 = 112 nM T18477 CI1G9X 137638702 IC50 = 14 nM T18477 CU4ZQ2 137638985 IC50 = 514 nM T18477 C4Q9JZ 137640085 IC50 = 749 nM T18477 C21FBO 137640720 IC50 = 28 nM T18477 CV0E9Z 137641466 IC50 = 473 nM T18477 CS3KF0 137642154 Ki = 1230 nM T18477 C12MZJ 137645122 IC50 = 260 nM T18477 C5CQ9Z 137645320 IC50 = 154 nM T18477 CPT60O 137645600 IC50 = 189 nM T18477 CHR4Z3 137648200 IC50 = 752 nM T18477 CJ16QN 137649039 IC50 = 151 nM T18477 CX4QS7 137649776 IC50 = 368 nM T18477 CF3L0U 137649852 IC50 = 836 nM T18477 CNXW27 137650729 IC50 = 285 nM T18477 CJ39SV 137650769 IC50 = 429 nM T18477 CL5J0D 137651203 IC50 = 206 nM T18477 CBTS61 137651332 IC50 > 10000 nM T18477 CQA9I8 137651592 IC50 = 98 nM T18477 CU9X3H 137651850 IC50 = 72 nM T18477 C7NG3S 137653255 IC50 = 21 nM T18477 C56PSW 137653748 IC50 = 397 nM T18477 CCEA75 137654206 IC50 = 122 nM T18477 C06UCI 137654541 IC50 = 106 nM T18477 C9YPV6 137657005 IC50 = 206 nM T18477 CBUZ81 137657937 IC50 = 79 nM T18477 C2A8IQ 137657990 IC50 > 10000 nM T18477 CA7G0C 137658950 IC50 = 39 nM T18477 COR37X 137659330 IC50 > 1000 nM T18477 CPH71E 137659954 IC50 = 407 nM T18477 CO6XK1 137660391 Ki = 184 nM T18477 C9SC4G 137660536 IC50 = 259 nM T18477 C43OWV 145953418 IC50 = 40 nM T18477 CNE6Q7 145953506 IC50 > 1000 nM T18477 CU9J0X 145954267 IC50 > 1000 nM T18477 CROY34 145956057 IC50 = 260 nM T18477 C9CBZ7 145956245 IC50 = 84.8 nM T18477 C14ICP 145956607 IC50 = 100 nM T18477 CG5IT7 145956784 IC50 > 1000 nM T18477 C20VAD 145957128 IC50 = 370 nM T18477 CR26HS 145959950 IC50 = 123 nM T18477 CWU27Z 145969804 IC50 > 100000 nM T18477 C63KEL 145970838 IC50 = 20200 nM T18477 C7UG3O 145971121 IC50 > 100000 nM T18477 CGSA67 145971928 IC50 = 47 nM T18477 CDVM26 145971994 IC50 > 1000 nM T18477 C9VDE5 145982499 IC50 = 40.2 nM T18477 C6OL1K 145983267 IC50 = 55.9 nM T18477 C8O1GU 145983616 IC50 = 49.3 nM T18477 C17UTC 145983813 IC50 = 85.7 nM T18477 CIWO70 145984314 IC50 = 52.1 nM T18477 C9ZKC1 145984665 IC50 = 58.6 nM T18477 CN6KB9 145985243 IC50 = 46.3 nM T18477 C0DR4V 146034184 IC50 = 21 nM T18477 CKO79M 155511775 IC50 = 70 nM T18477 CQ5L3O 155515228 IC50 = 52670 nM T18477 C0ZY8Q 155516833 IC50 > 100000 nM T18477 CEG67W 155518415 IC50 = 54680 nM T18477 C9AC7B 155518571 IC50 = 164 nM T18477 CDY5H6 155519645 IC50 = 77210 nM T18477 C83HYP 155521152 IC50 = 430 nM T18477 C6Q4LC 155521952 IC50 = 15290 nM T18477 CJ34YH 155524691 IC50 = 643 nM T18477 C68ZRJ 155524949 IC50 = 97.11 nM T18477 CQ3AI0 155525851 IC50 = 302290 nM T18477 CX2D6L 155525906 IC50 = 1702 nM T18477 CH52FD 155526273 IC50 > 1000000 nM T18477 CU4X5I 155527383 IC50 > 10000 nM T18477 C9O0EU 155528011 IC50 = 72 nM T18477 CLVW69 155528303 IC50 > 1000000 nM T18477 C5F1IZ 155528743 IC50 > 1000000 nM T18477 C9TIO5 155528896 IC50 = 169340 nM T18477 C1B2FN 155530610 IC50 = 145800 nM T18477 C0VZ9J 155532068 IC50 > 1000000 nM T18477 CVL8J4 155532571 IC50 = 280 nM T18477 C6LTV0 155536018 IC50 = 42980 nM T18477 C45YWP 155537090 IC50 = 52.97 nM T18477 C8WNG3 155539047 IC50 = 60 nM T18477 CLD19W 155539311 IC50 = 153070 nM T18477 C9PFH1 155539933 IC50 = 13620 nM T18477 CNC1O0 155543432 IC50 = 89830 nM T18477 CFM68U 155545469 IC50 > 1000 nM T18477 CWZ82Y 155546946 IC50 = 1258 nM T18477 CE9R1Q 155549076 IC50 = 76810 nM T18477 C02YXA 155550058 IC50 = 186070 nM T18477 CUN7G5 155554476 IC50 = 8.319 nM T18477 CTC6O0 155554826 IC50 > 10000 nM T18477 CVH3K6 155555734 IC50 = 630 nM T18477 CG7OQ2 155556818 IC50 > 1000 nM T18477 CE1Q6X 155558343 IC50 = 58 nM T18477 CMPA40 155559139 IC50 = 204 nM T18477 CG0HE7 155559221 IC50 = 6200 nM T18477 C3QA1U 155561308 IC50 = 150 nM T18477 C8R0WI 155561564 IC50 = 67060 nM T18477 C8JD0L 155561717 IC50 = 36620 nM T18477 C7L2RV 155562486 IC50 = 67 nM T18477 C1JQG6 155563956 IC50 = 1506 nM T18477 C0XJ5Q 155564241 IC50 = 22630 nM T18477 C40KVW 155565004 IC50 = 42410 nM T18477 C3J4AQ 155567472 IC50 > 10000 nM T18477 C3IU9Q 155567695 IC50 = 87 nM T18477 D05NWF 6022 EC50 = 120000 nM T18477 D07APP 131255 EC50 > 50000 nM T18477 D07TYL 1130 IC50 = 12500 nM T18477 D08OLB 49784944 IC50 = 3000 nM T18477 D0C2UJ 8974 IC50 <= 1250000 nM T18477 D0K0TJ 24772860 Ki = 4 nM T18477 D0T4MS 4369536 IC50 = 25 nM T18477 D0ZA6G 6323491 IC50 = 150 nM T72835 D02AUB 9811353 IC50 > 500000 nM T72835 CKM1X8 128677 IC50 = 50 nM T72835 C1GDY7 587790 IC50 = 31700 nM T72835 C96KNY 643990 IC50 = 300000 nM T72835 CXI3Y4 645569 IC50 > 100000 nM T72835 C5Q0FP 745480 IC50 = 49000 nM T72835 CYBV18 916176 IC50 = 27000 nM T72835 C16YNJ 962611 IC50 = 95000 nM T72835 COB6U4 2807642 IC50 = 3000 nM T72835 CYBK67 5481003 IC50 = 6600 nM T72835 CT3BF9 9797597 IC50 = 88 nM T72835 C74QCT 9798233 IC50 = 60 nM T72835 CCI90K 9799728 IC50 = 620 nM T72835 C18UGE 9818339 IC50 = 8400 nM T72835 CJQ2W6 9835897 IC50 > 1000 nM T72835 C6G5RT 9836507 IC50 > 4000 nM T72835 CUGN49 9836683 IC50 = 70 nM T72835 CJ5SU0 9839311 IC50 = 20 nM T72835 CSK6P4 9841875 IC50 = 500 nM T72835 C5DRX6 9856682 IC50 = 60 nM T72835 C9MA3Z 9858009 IC50 = 16 nM T72835 C0ZQV7 9858022 IC50 = 43 nM T72835 C3MG0X 9860649 IC50 = 690 nM T72835 C8IO4M 9878726 IC50 = 42000 nM T72835 C91VCO 9878930 IC50 = 20 nM T72835 CP34JF 9879093 IC50 = 600 nM T72835 C5S6CZ 9879529 IC50 = 6 nM T72835 CBKH73 9880710 IC50 = 100 nM T72835 C1L5WE 9880711 IC50 = 31 nM T72835 C0O5BM 9881984 IC50 = 2200 nM T72835 C0W1SB 9882382 IC50 = 660 nM T72835 CY7KG3 9883504 IC50 = 8 nM T72835 CL1FR4 9900816 IC50 = 1 nM T72835 C3D1XN 9900943 IC50 = 150 nM T72835 C9DHR2 9901085 IC50 = 800 nM T72835 CRND31 9901574 IC50 = 170 nM T72835 CBM7Y3 9903965 IC50 = 1800 nM T72835 CKJ7T0 9903998 IC50 = 22000 nM T72835 C1JI7S 9904207 IC50 = 4000 nM T72835 C3VJ9K 9904395 IC50 = 140 nM T72835 C62JUP 9904430 IC50 > 4000 nM T72835 CYN51E 9905179 IC50 = 12 nM T72835 CDML85 9906347 IC50 = 4 nM T72835 CO63ID 9921367 IC50 = 1700 nM T72835 CQ4WG3 9921987 IC50 = 100 nM T72835 C9T3ME 9922373 IC50 = 45 nM T72835 CO5L2R 9922793 IC50 = 76 nM T72835 C36KVQ 9922943 IC50 = 150 nM T72835 CW5P9J 9924766 IC50 = 100 nM T72835 C7QP1H 9944101 IC50 = 30 nM T72835 C2JZW5 9944163 IC50 = 55 nM T72835 C9AJP0 9944774 IC50 = 130 nM T72835 CL9I6U 9945784 IC50 = 19 nM T72835 CB3P7T 9946091 IC50 > 1000 nM T72835 CYJ59B 9946991 IC50 = 9 nM T72835 CAFK13 9947244 IC50 = 5 nM T72835 CR4LP3 9948282 IC50 = 16000 nM T72835 CNH47D 9948311 IC50 = 3200 nM T72835 C0YEQ7 9952465 IC50 = 120 nM T72835 C2TYQ1 9953413 IC50 > 100000 nM T72835 CWH3L0 9965679 IC50 = 20 nM T72835 CI4DU5 9966679 IC50 = 32 nM T72835 CFEI36 9967126 IC50 = 79 nM T72835 CA5W9Z 9967290 IC50 = 670 nM T72835 CS9DM3 9967511 IC50 = 340 nM T72835 CYXW91 9968489 IC50 = 44 nM T72835 CZ98HT 9977686 IC50 > 500000 nM T72835 CX30HT 10089338 IC50 = 0.7 nM T72835 C8TZ5Q 10101726 IC50 = 30000 nM T72835 C4E8NU 10106199 IC50 = 3300 nM T72835 COIF97 10107659 IC50 = 1400 nM T72835 CY23GM 10108997 IC50 = 200 nM T72835 C2P4UO 10110987 IC50 > 4000 nM T72835 CTW3P9 10116693 IC50 = 110 nM T72835 C07COW 10132518 IC50 = 80 nM T72835 C6N1FU 10134148 IC50 > 4000 nM T72835 CH49BD 10154440 IC50 = 630 nM T72835 COF2S9 10154441 IC50 = 20 nM T72835 CL7H2B 10154801 IC50 = 210 nM T72835 C0CP1T 10155661 IC50 = 300 nM T72835 CSB5F9 10156828 IC50 = 110 nM T72835 CF4DP2 10177047 IC50 = 60 nM T72835 C6RN4F 10178848 IC50 = 6 nM T72835 CHN3X1 10202790 IC50 > 4000 nM T72835 CD95KA 10221525 IC50 = 520 nM T72835 CJZU30 10267771 IC50 = 13 nM T72835 C2OQ0K 10267925 IC50 = 370 nM T72835 C9C0UG 10291112 IC50 > 4000 nM T72835 CWZU32 10291698 IC50 = 31 nM T72835 CTUP45 10291904 IC50 > 4000 nM T72835 CM05NG 10298900 IC50 = 120 nM T72835 C7KO6U 10361323 IC50 = 7 nM T72835 C1NX9Z 10469899 IC50 < 30000 nM T72835 CZ3DK8 10566084 IC50 = 17000 nM T72835 C5Q8EF 10566766 IC50 = 15000 nM T72835 CN3H5M 10632359 IC50 = 250 nM T72835 C6QZG3 10686899 IC50 > 4000 nM T72835 CZF1H3 10708446 IC50 = 200 nM T72835 CAPG02 10732433 IC50 > 1000 nM T72835 C6K5GC 10860379 IC50 = 21 nM T72835 CSO95L 10862219 IC50 = 864 nM T72835 C7OFZ9 10863087 IC50 = 120 nM T72835 C6PRJ8 10880644 IC50 = 35 nM T72835 C2VX3P 10886395 IC50 > 100000 nM T72835 CV9I3D 10891751 IC50 = 3 nM T72835 C9X6VP 10892285 IC50 = 940 nM T72835 C9DUB8 10892642 IC50 = 8 nM T72835 CS1T3C 10896625 IC50 = 115 nM T72835 CARC06 10904579 IC50 = 150 nM T72835 CHWL69 10905666 IC50 = 25 nM T72835 CLPA31 10906508 IC50 = 34 nM T72835 C7YG6L 10924566 IC50 = 28 nM T72835 CR51AV 10970154 IC50 = 4 nM T72835 CQ6E7Y 10970207 IC50 > 1000 nM T72835 CB31OE 10980658 IC50 = 870 nM T72835 C94UAC 10982608 IC50 = 4 nM T72835 CVR4Y3 11001541 IC50 = 25 nM T72835 CCP7K5 11013542 IC50 = 5 nM T72835 C1ZRL6 11014018 IC50 = 5 nM T72835 CIW6J5 11023935 IC50 = 13 nM T72835 C7NCE4 11036406 IC50 = 2 nM T72835 CM5HI8 11045962 IC50 = 6 nM T72835 C7U2JK 11048059 IC50 = 28 nM T72835 C7E6GN 11048585 IC50 = 600 nM T72835 CNHY70 11057712 IC50 = 35 nM T72835 COE6W0 11068095 IC50 = 2 nM T72835 C9Q0MP 11070710 IC50 = 650 nM T72835 CZSV01 11078679 IC50 = 470 nM T72835 C1KE2T 11079237 IC50 = 7 nM T72835 C8SRX4 11080157 IC50 > 715 nM T72835 C5T1BO 11089640 IC50 = 5 nM T72835 CQYV18 11091464 IC50 = 770 nM T72835 CSF94U 11102008 IC50 = 830 nM T72835 C51PTF 11109642 IC50 = 18 nM T72835 C8RF0J 11111846 IC50 > 1000 nM T72835 C8WI4X 11120977 IC50 = 380 nM T72835 CUGV75 11122788 IC50 > 1000 nM T72835 CHIT70 11134430 IC50 = 43 nM T72835 CRPC48 11134652 IC50 = 680 nM T72835 C4Z0FP 11258464 IC50 = 41900 nM T72835 CKHO40 11558561 IC50 > 50000000 nM T72835 CN5M7E 11680708 IC50 > 50000000 nM T72835 C5DUF4 11760748 IC50 = 110 nM T72835 CF7GU9 11777631 IC50 < 30000 nM T72835 C8BJ0L 11783098 IC50 = 180 nM T72835 C43LZD 11783922 IC50 = 870 nM T72835 CKRM28 11793014 IC50 > 1000 nM T72835 CLX8Z9 11825588 IC50 = 5 nM T72835 C7SG8X 11828434 IC50 = 2.8 nM T72835 C62DAO 16114614 IC50 = 800 nM T72835 C1ET3V 16114615 IC50 = 1000 nM T72835 CQ90BS 16114616 IC50 = 3300 nM T72835 CA4MJ7 16114618 IC50 = 8400 nM T72835 CWGO19 16114619 IC50 = 1300 nM T72835 CTC76N 16114620 IC50 = 8400 nM T72835 CM7Z2R 16115893 IC50 > 500000 nM T72835 C41WNZ 16116039 IC50 = 4900 nM T72835 CUE4D8 16116040 IC50 = 85400 nM T72835 C2EHS8 16116042 IC50 = 18700 nM T72835 CTG1J6 16116159 IC50 = 2300 nM T72835 CZH0G1 16116162 IC50 = 8700 nM T72835 C5GZB3 16116163 IC50 > 500000 nM T72835 CKI2E4 16116165 IC50 = 52400 nM T72835 C5Q4GR 16116166 IC50 > 500000 nM T72835 C7F1DY 16116286 IC50 = 48600 nM T72835 CU4OF0 16116421 IC50 > 500000 nM T72835 C89WXF 16116422 IC50 > 500000 nM T72835 C82KGR 16116555 IC50 > 500000 nM T72835 C9DME7 16116556 IC50 = 57200 nM T72835 CU2IB8 16116557 IC50 = 132000 nM T72835 CTXB17 16116558 IC50 > 500000 nM T72835 CFU0D9 16116559 IC50 = 113700 nM T72835 C7WJ0Y 16725848 IC50 = 9700 nM T72835 C5WSK1 23669281 IC50 = 3100 nM T72835 CC12EZ 23709469 IC50 = 280000 nM T72835 C36WMA 44264201 IC50 > 4000 nM T72835 CU30LF 44285871 IC50 = 10000000 nM T72835 C94VZY 44285873 IC50 = 8000000 nM T72835 C4J3NI 44285918 IC50 > 10000000 nM T72835 C7Y2QI 44285932 IC50 > 10000000 nM T72835 CXDS56 44285933 IC50 = 3000000 nM T72835 C4LNK6 44286072 IC50 = 1600000 nM T72835 CPW18X 44286163 IC50 = 6700000 nM T72835 C3KEI4 44286164 IC50 = 6000000 nM T72835 CU6T4G 44286241 IC50 = 7000000 nM T72835 C57VYM 44286390 IC50 = 6000000 nM T72835 CHF78N 44286451 IC50 = 7000000 nM T72835 CQP9G7 44304820 IC50 > 1000000 nM T72835 C5PC9B 44314807 IC50 = 2800000 nM T72835 C8V5HM 44314808 IC50 = 600000 nM T72835 C9YI8T 44314810 IC50 = 360000 nM T72835 C9FOU7 44314839 IC50 = 300000 nM T72835 C4FE2A 44314950 IC50 = 3000000 nM T72835 CMR6V4 44314968 IC50 = 3000000 nM T72835 C7S8PZ 44314993 IC50 > 2500000 nM T72835 CG2R9Y 44314996 IC50 > 2500000 nM T72835 CH5N4J 44315249 IC50 > 4000000 nM T72835 CZ06IY 44315261 IC50 = 3000000 nM T72835 C6JB5F 44315289 IC50 = 840000 nM T72835 CJN5S6 44315290 IC50 = 530000 nM T72835 CE18QO 44315291 IC50 = 950000 nM T72835 C7J8LN 44315330 IC50 = 350000 nM T72835 CECK48 44315332 IC50 > 10000000 nM T72835 CH40ER 44325713 IC50 = 500000 nM T72835 CB14NL 44325784 IC50 = 50000 nM T72835 CO3WB1 44325797 IC50 = 500000 nM T72835 CWCI90 44325812 IC50 = 1000000 nM T72835 CI6W5K 44325824 IC50 = 100000 nM T72835 C5ZGP4 44325830 IC50 = 100000 nM T72835 CX1PZ3 44325844 IC50 = 300000 nM T72835 C5FP7T 44325913 IC50 = 3000000 nM T72835 CH0YQ4 44325932 IC50 = 5000000 nM T72835 CC0DP9 44325956 IC50 = 900000 nM T72835 C4EQ5L 44325958 IC50 = 500000 nM T72835 CD1Y6W 44340382 IC50 > 1000000 nM T72835 CC7G9J 44340394 IC50 > 1000000 nM T72835 C2Q7LW 44340567 IC50 > 1000000 nM T72835 CZG4T2 44340638 IC50 > 1000000 nM T72835 CK1GA0 44340639 IC50 > 1000000 nM T72835 CM7P9U 44344139 IC50 = 13 nM T72835 CICW90 44356343 IC50 = 160000 nM T72835 C1VH5G 44356439 IC50 > 500000 nM T72835 CK7WE9 44356515 IC50 > 500000 nM T72835 CPM04F 44356616 IC50 > 500000 nM T72835 C8CR4F 44356617 IC50 > 500000 nM T72835 CL8M6C 44360868 IC50 > 10000000 nM T72835 C02ULA 44360870 IC50 > 10000000 nM T72835 CXK84H 44360912 IC50 > 10000000 nM T72835 CXL0S8 44387278 IC50 > 1000000 nM T72835 CIAL79 44387290 IC50 > 1000000 nM T72835 CHIF62 44387291 IC50 > 1000000 nM T72835 C6FK5A 44387293 IC50 = 240000 nM T72835 C7WPK9 44387294 IC50 = 360000 nM T72835 CPQ09T 44387295 IC50 > 1000000 nM T72835 CPT5K3 44387297 IC50 > 1000000 nM T72835 CS0M3D 44399068 IC50 > 50000000 nM T72835 C67QAL 44399069 IC50 > 50000000 nM T72835 C3TJ5S 44399147 IC50 > 50000000 nM T72835 CB74WV 44399232 IC50 > 50000000 nM T72835 CVDP57 44399253 IC50 > 50000000 nM T72835 C0ZIP8 44420653 IC50 = 3000 nM T72835 C5QXG3 44420654 IC50 = 3100 nM T72835 C2S9CH 44420657 IC50 = 61400 nM T72835 C8Y1HG 44420659 IC50 = 48000 nM T72835 CQ08EK 44420661 IC50 = 15700 nM T72835 CA9T5O 44420662 IC50 > 500000 nM T72835 C7F6HB 44456838 IC50 = 600000 nM T72835 CZG86H 44456859 IC50 = 1000000 nM T72835 CW8KR3 46845959 IC50 = 2500000 nM T72835 C8MUB4 46881482 IC50 = 11000000 nM T72835 CM2TE6 46881483 IC50 = 5000000 nM T72835 CE7OJ4 46881484 IC50 = 3000000 nM T72835 CS68ZT 46881485 IC50 = 5000000 nM T72835 COJ35S 46881517 IC50 = 15000000 nM T72835 C8Q0YB 46881518 IC50 = 6000000 nM T72835 C1RN8P 53323826 IC50 > 10000000 nM T72835 CK9Q2E 56675135 IC50 = 32000 nM T72835 C0BAV1 70687644 IC50 = 41000 nM T72835 C0MZH5 70687646 IC50 = 49000 nM T72835 CVM5H6 70689898 IC50 = 24000 nM T72835 CJA84B 70696227 IC50 = 1125000 nM T72835 CS1FC2 71450419 IC50 = 5460000 nM T72835 CEPH60 71452644 IC50 > 1000000 nM T72835 CN0ZI6 71458017 IC50 > 1000000 nM T72835 CGE8R2 71715994 IC50 = 16000 nM T72835 C7E0WX 71715999 IC50 = 2100000 nM T72835 C0FR3U 71716010 IC50 = 3500 nM T72835 C3S7VA 71716029 IC50 = 1000000 nM T72835 C3JQ6N 71716030 IC50 = 500000 nM T72835 CEO6H7 71716031 IC50 = 3200000 nM T72835 C6C0ZR 71716033 IC50 = 2000000 nM T72835 CHJ5U3 71716622 IC50 > 6600000 nM T72835 CJ2Q9U 71716626 IC50 = 1500000 nM T72835 C2RAX0 71716634 IC50 = 20000000 nM T72835 C1B3SM 71717205 IC50 > 10000000 nM T72835 C6IM8H 71717206 IC50 = 500000 nM T72835 CO9E1I 71717225 IC50 = 80000 nM T72835 CK27AE 71717234 IC50 = 1000000 nM T72835 CGQB06 71717239 IC50 = 20000000 nM T72835 CY37OD 71717829 IC50 = 1000000 nM T72835 CWQ63V 71717841 IC50 = 1400000 nM T72835 C8P0KB 71717843 IC50 = 2000000 nM T72835 C7NA8Z 71717847 IC50 = 20200000 nM T72835 C9BQW5 71717848 IC50 = 4600000 nM T72835 C1N3RG 71718477 IC50 > 6600000 nM T72835 C8KT6Z 71718487 IC50 = 36000000 nM T72835 CL25WA 71718488 IC50 = 6100000 nM T72835 CCO93Y 71719057 IC50 = 330000 nM T72835 CH42FQ 71719059 IC50 = 300000 nM T72835 CBLP16 71719067 IC50 = 4900000 nM T72835 C8MHG7 71719069 IC50 = 34400000 nM T72835 CQR6H7 71719671 IC50 = 500000 nM T72835 C2XBN3 71719672 IC50 = 400000 nM T72835 CF85XK 71719677 IC50 = 32000000 nM T72835 CPK9T0 71719678 IC50 = 11500000 nM T72835 C97AXO 71719679 IC50 = 14600000 nM T72835 CXZA30 71720268 IC50 = 2000000 nM T72835 C32CAX 71720271 IC50 = 4000000 nM T72835 CSMU14 71720272 IC50 = 5000000 nM T72835 C7XR6V 71720274 IC50 = 2500000 nM T72835 C23OXT 71720283 IC50 = 14000000 nM T72835 CTHW87 71720284 IC50 = 8000000 nM T72835 CCNR81 71720285 IC50 = 20000000 nM T72835 CGYI26 71720286 IC50 = 9500000 nM T72835 C53BRY 71720287 IC50 = 2600000 nM T72835 CP71RD 71720288 IC50 = 7000000 nM T72835 CL50FA 73351434 IC50 = 300000 nM T72835 CEH94N 73352890 IC50 = 80000 nM T72835 C3FIJ8 73354415 IC50 = 300000 nM T72835 CBCN75 73355970 IC50 = 2900000 nM T72835 C6MGQ0 73355972 IC50 = 1000000 nM T72835 C8TE5P 76335199 IC50 = 280000 nM T72835 CQ1W3X 90663369 IC50 = 16000000 nM T72835 C6CYV1 90664029 IC50 = 500000 nM T72835 CIU4H8 90664107 IC50 = 5000000 nM T72835 CO2DA9 90664124 IC50 = 600000 nM T72835 CKZP37 90664125 IC50 > 1000000 nM T72835 C1TG5J 90664143 IC50 = 350000 nM T72835 CJ63KL 90664145 IC50 > 10000000 nM T72835 C2QW4L 90664147 IC50 > 10000000 nM T72835 CM4V1J 90664149 IC50 > 10000000 nM T72835 CNQZ02 90664151 IC50 = 80000 nM T72835 CV8B6I 90664153 IC50 = 15800000 nM T72835 CL37TX 90664156 IC50 = 3800000 nM T72835 CXN0Q3 90664160 IC50 = 280000 nM T72835 C86TFW 90664161 IC50 = 650000 nM T72835 C7V9EN 90664162 IC50 = 590000 nM T72835 C5ZKM2 90664163 IC50 > 1000000 nM T72835 CMZK65 90664164 IC50 = 5000000 nM T72835 C2J7FQ 90664165 IC50 = 1000000 nM T72835 C49RXN 90664166 IC50 = 1150000 nM T72835 CUWF73 90664170 IC50 = 700000 nM T72835 CE1DY2 90664171 IC50 = 900000 nM T72835 C13WQJ 90664172 IC50 = 270000 nM T72835 C6VS3D 90664191 IC50 = 10000 nM T72835 CO85IQ 90664193 IC50 = 30000 nM T72835 C90MHO 90664197 IC50 = 60000 nM T72835 C84CFR 90664199 IC50 = 37000 nM T72835 C1NKI3 90664201 IC50 = 1500 ug.mL-1 T72835 C9XAE4 90664202 IC50 = 100 ug.mL-1 T72835 CBI07N 90664204 IC50 = 30000 nM T72835 CKIU49 90664206 IC50 = 200000 nM T72835 CDVW23 90664222 IC50 = 700000 nM T72835 CJ4FT2 90664262 IC50 = 700000 nM T72835 CJ3O0E 90664264 IC50 = 3500 nM T72835 C6KN7R 90664265 IC50 > 100000 nM T72835 CF9XM7 118714544 IC50 = 2080000 nM T72835 CZU9S3 118714545 IC50 = 140000 nM T72835 C6G1LI 118714546 IC50 = 220000 nM T72835 CIF1K3 118714547 IC50 = 76000 nM T72835 CDYU78 118718895 IC50 = 4300 nM T72835 C1A5QG 118718900 IC50 = 13000 nM T72835 CK6Q9M 118718901 IC50 = 1500 nM T72835 C15YGB 118719302 IC50 > 1000000 nM T72835 CI3VJ0 118719304 IC50 > 100000 nM T72835 CZH6T3 118719305 IC50 > 1000000 nM T72835 C4BGF1 118719306 IC50 > 100000 nM T72835 C2FX6G 135506443 IC50 = 20000 nM T72835 D0E9NT 11874 IC50 > 500000 nM T72835 D0Y3TZ 370 IC50 > 500000 nM T32973 CI0DG1 764318 IC50 = 180 nM T32973 CPA63I 3107941 Ki = 105 nM T32973 C6SO2K 3708081 IC50 = 170 nM T32973 CRT04P 44298904 IC50 = 31 nM T32973 CCLG83 44298942 IC50 = 55 nM T32973 CVE6Z8 44299051 IC50 = 1000 nM T32973 CLC74A 44299052 IC50 = 38 nM T32973 C3DRB6 45496892 IC50 = 160 nM T32973 CU3WO1 90656770 IC50 = 140 nM T32973 CUZ5D8 90656771 IC50 = 192 nM T32973 CA0I4Q 90656772 IC50 = 108 nM T32973 CHD13U 90656773 IC50 = 282 nM T32973 C7CZK1 90656774 IC50 = 138 nM T32973 CMBD94 90656775 IC50 = 18 nM T32973 CH1LG5 90656776 IC50 = 49 nM T32973 C9YW4M 90656777 IC50 = 28 nM T32973 C0YFV2 90656778 IC50 = 169 nM T32973 C4BNV6 90656779 IC50 = 49 nM T32973 C8GMB3 90656780 IC50 = 97 nM T32973 C6ZT9S 90656781 IC50 = 83 nM T32973 C4LC5K 90656782 IC50 = 348 nM T32973 CV0ZW9 90656783 IC50 = 60 nM T32973 CS83DE 90656784 IC50 = 5 nM T32973 CC0HQ5 90656785 IC50 = 79 nM T32973 C6RU7O 90656786 IC50 = 29 nM T32973 CIY4S9 90656787 IC50 = 11 nM T32973 C01DTE 90656788 IC50 = 41 nM T32973 CV98QR 90656789 IC50 = 9 nM T32973 C5UV6T 90656790 IC50 = 124 nM T32973 C9O6FJ 90656791 IC50 = 1640 nM T32973 CN7BQ9 90656792 IC50 = 65 nM T32973 C2O9IM 90656793 IC50 = 15 nM T32973 C0U3KA 90656794 IC50 = 41 nM T32973 C0AZ6Q 90656795 IC50 = 3.2 nM T32973 C89FRT 90656797 IC50 = 7.8 nM T32973 CFB02X 90656798 IC50 = 343 nM T32973 C6E0RT 90656799 IC50 = 9 nM T32973 CV04JO 127037715 IC50 = 71 nM T32973 C6MQI3 127038634 IC50 > 10000 nM T32973 CM1CO8 127038635 IC50 = 356 nM T32973 C3WYE0 127038636 IC50 > 10000 nM T32973 CW6F1G 127038637 IC50 = 128 nM T32973 C09UKF 127038638 IC50 = 2259 nM T32973 C8JGW4 127038639 IC50 = 1035 nM T32973 CO7I3Q 127038645 IC50 > 10000 nM T32973 CBIQ30 127038646 IC50 = 323 nM T32973 CDO09Y 127038719 IC50 = 73 nM T32973 C38JYQ 127038989 IC50 = 1459 nM T32973 CC2O5W 127038990 IC50 = 252 nM T32973 C5VE8N 127038991 IC50 = 6296 nM T32973 CW89HP 127038992 IC50 = 1359 nM T32973 C8Z3HL 127039269 IC50 = 882 nM T32973 CU57WL 127039270 IC50 = 5050 nM T32973 C4JR2O 127039271 IC50 = 5854 nM T32973 C3FYV7 127039330 IC50 = 9249 nM T32973 CA9I0O 127039395 IC50 = 269 nM T32973 C2EX1W 127039396 IC50 > 10000 nM T32973 CH7P9N 127039594 IC50 = 4384 nM T32973 CGY9L1 127039595 IC50 = 7749 nM T32973 C7QP0E 127039715 IC50 = 282 nM T32973 C1MN6H 127039716 IC50 > 10000 nM T32973 C65YMT 127039717 IC50 = 332 nM T32973 CV3DF7 127039734 IC50 = 67 nM T32973 CQ69EI 127039735 IC50 = 23 nM T32973 CUQ5H2 127039930 IC50 > 10000 nM T32973 C4B3JS 127039931 IC50 > 10000 nM T32973 CN73ZO 127039932 IC50 = 3889 nM T32973 CJ9IQ8 127040049 IC50 > 10000 nM T32973 C8RPF9 127040057 IC50 = 49 nM T32973 C63WGY 127040119 IC50 = 6 nM T32973 C5Y8BK 127040330 IC50 = 1086 nM T32973 C1PR6T 127040663 IC50 > 10000 nM T32973 CKS4F0 127040664 IC50 = 6745 nM T32973 C9P4CX 127040726 IC50 = 33 nM T32973 C5G2EC 127040909 IC50 > 10000 nM T32973 CH1FG6 127040984 IC50 = 2272 nM T32973 CL9DB6 127040985 IC50 = 1818 nM T32973 C8Y3RC 127040986 IC50 > 10000 nM T32973 CF23HM 127040987 IC50 > 10000 nM T32973 CSF23D 127041612 IC50 = 425 nM T32973 CE5N9Z 127041613 IC50 = 601 nM T32973 CD8BP0 127041614 IC50 > 10000 nM T32973 CD2XR0 127041615 IC50 = 378 nM T32973 CO0NJ1 127041616 IC50 = 5854 nM T32973 C5DKU9 127041617 IC50 = 586 nM T32973 CEHK53 127041618 IC50 > 10000 nM T32973 CEL1O2 127041744 IC50 = 169 nM T32973 C9Q8DT 127041745 IC50 = 93 nM T32973 C9JOV0 127041985 IC50 = 593 nM T32973 CH19UD 127042050 IC50 = 121 nM T32973 CJ27CG 127042051 IC50 = 6 nM T32973 CVE08P 127042052 IC50 = 73 nM T32973 CIE83Y 127042053 IC50 = 969 nM T32973 CAT46D 127042341 IC50 = 12 nM T32973 CN1M5T 127042410 IC50 > 10000 nM T32973 CO2IY7 127042411 IC50 = 33 nM T32973 CW2F7T 127042682 IC50 = 47 nM T32973 CZ3BE8 127042683 IC50 = 35 nM T32973 CD42KE 127042684 IC50 = 45 nM T32973 C2C9DK 127042738 IC50 = 32 nM T32973 C36SAQ 127042739 IC50 = 71 nM T32973 CNTF18 127042740 IC50 = 5 nM T32973 C1F2AW 155512129 IC50 = 34 nM T32973 CPJK82 155512819 IC50 = 82 nM T32973 C5OGP9 155513654 IC50 = 0.26 nM T32973 CBGY41 155515971 IC50 = 59 nM T32973 C64OMX 155518715 IC50 = 18 nM T32973 C5KH2Y 155523364 IC50 = 7.1 nM T32973 CGI0C3 155529023 IC50 = 15 nM T32973 C6F1JL 155532513 IC50 = 280 nM T32973 CETH73 155533920 IC50 = 9.8 nM T32973 C03EVD 155535966 IC50 = 5.5 nM T32973 C67DMO 155536395 IC50 = 15 nM T32973 C3BWI8 155537675 IC50 = 3.6 nM T32973 CKR9O0 155540299 IC50 = 10 nM T32973 CTG0X5 155540609 IC50 = 12 nM T32973 CZT36F 155541834 IC50 = 290 nM T32973 CW5IN2 155542032 IC50 = 33 nM T32973 CMV89O 155544241 IC50 = 160 nM T32973 CKZI03 155549215 IC50 = 78 nM T32973 C6IQO0 155550525 IC50 = 26 nM T32973 CS35NF 155550740 IC50 = 1.3 nM T32973 C2B7KY 155552502 IC50 = 1.4 nM T32973 CL40SZ 155553142 IC50 = 0.12 nM T32973 C3ZO7Y 155556864 IC50 = 870 nM T32973 CF5HV2 155557380 IC50 = 0.47 nM T32973 C2IUT6 155558910 IC50 > 10000 nM T32973 CQ08FY 155562629 IC50 = 110 nM T32973 C54SNK 155567233 IC50 = 96 nM T32973 D0W6HI 90656796 IC50 = 0.9 nM T92689 D01BYB 5957 EC50 = 3300 nM T92689 D06ACW 6083 EC50 = 17250 nM T92689 D0H2UB 5361 Ki = 112.2 nM T92689 D0KE4Z 5310954 EC50 = 1500 nM T92689 D0Z7FU 6133 EC50 > 100000 nM T92689 CPQ81V 171069 EC50 = 4500 nM T92689 CCJ8P0 440317 EC50 = 63.1 nM T92689 C18IQO 10080003 Ki = 7585.78 nM T92689 C04CWB 10080210 Ki = 1000 nM T92689 CA8GR7 10080218 Ki = 446.68 nM T92689 C3L6KW 10994891 EC50 = 17250 nM T92689 CHB3C7 11510273 Ki > 15000 nM T92689 CT74ZJ 11560464 Ki > 15000 nM T92689 CGQV15 11564436 Ki = 107.15 nM T92689 CUD1J5 11611428 Ki > 15000 nM T92689 CX7J8F 11636756 Ki = 44.67 nM T92689 C10PSW 11679780 Ki = 2398.83 nM T92689 CQ40BH 14753886 EC50 = 900 nM T92689 CCZ8N0 16155349 Ki = 75.86 nM T92689 CN4BT9 16163319 Ki = 302 nM T92689 C56DVM 23656757 EC50 = 478.63 nM T92689 CM45HO 23656759 EC50 = 1288.25 nM T92689 CQ46IG 44353592 EC50 = 7000 nM T92689 C30CIT 49856886 EC50 = 13000 nM T92689 CJ2RM6 56673378 EC50 >= 40000 nM T92689 C4VFI2 68530100 Ki > 15000 nM T92689 CJK95G 71450314 EC50 = 2900 nM T92689 CL0X8W 73347374 EC50 = 1400 nM T92689 CLXM46 73351984 EC50 = 1000 nM T92689 C9CWV3 73353445 EC50 = 130 nM T92689 C1AJ6L 73354953 EC50 = 1500 nM T92689 CAS84P 76324375 EC50 > 100000 nM T92689 C78INB 118725181 EC50 = 3680 nM T92689 CM8N4I 122195891 EC50 = 1000 nM T92689 CULF46 122195892 EC50 = 500 nM T92689 CC2JO4 122195893 EC50 = 1100 nM T92689 C9HK0N 122195894 EC50 = 900 nM T92689 CZ1XL2 122195895 EC50 = 1000 nM T92689 D05MXI 42611190 IC50 > 10000 nM T92689 D05NWF 6022 EC50 = 1700 nM T92689 D07MTB 11510579 Ki > 15000 nM T92689 D0B0ZQ 9875920 EC50 > 100000 nM T92689 D0D8CZ 15993 EC50 = 9000 nM T92689 D0U1OJ 5310983 EC50 = 50000 nM T92689 D0V4GQ 5310996 EC50 = 30000 nM T28484 D0X5SI 193653 IC50 > 63000 nM T28484 D02AAO 10368812 IC50 = 429 nM T28484 D04VWJ 44224257 IC50 = 6 nM T28484 D0L4VI 5862 IC50 > 63000 nM T28484 D0PW4N 6851740 IC50 = 1.2 nM T28484 D0Q5QC 23634407 IC50 = 8 nM T28484 D0W9SL 25167017 IC50 = 7 nM T28484 D0Z0HH 3503 IC50 = 25000 nM T28484 D02CXZ 57094730 Ki = 203 nM T28484 C8V5EI 9720 IC50 = 3200 nM T28484 CG9LF7 21261 IC50 > 63000 nM T28484 C6UFG1 23011 IC50 = 23000 nM T28484 C2AJZ0 37323 Ki = 200 nM T28484 CI5X0C 76044 Ki = 26 nM T28484 C8U9DP 83278 IC50 > 20000 nM T28484 C43JDE 99558 IC50 > 63000 nM T28484 CLN9B4 128239 IC50 = 55000 nM T28484 C19ZNI 207753 IC50 > 50000 nM T28484 CD54OR 215628 Ki = 1750 nM T28484 CB09MQ 246378 IC50 = 5600 nM T28484 CCLD38 262764 Ki = 150 nM T28484 CNVZ38 277164 Ki = 5230 nM T28484 CQ20WF 282773 IC50 = 25000 nM T28484 CT9MH5 283741 Ki = 2536.3 nM T28484 CON03C 303820 IC50 = 1000 nM T28484 C9WSY2 391237 EC50 < 30000 nM T28484 C31NSG 541056 IC50 = 2500 nM T28484 CCL43Q 613965 IC50 = 10000 nM T28484 C15QBR 675901 EC50 < 30000 nM T28484 C9CBS4 686905 IC50 = 493 nM T28484 CUR7M6 692940 EC50 = 20000 nM T28484 C2B9ZV 703864 EC50 < 30000 nM T28484 CI6N1Q 806204 EC50 = 3600 nM T28484 CJ4G8Y 806211 EC50 = 2200 nM T28484 CY3A5N 1049743 EC50 = 34000 nM T28484 CX7H0T 1190622 EC50 = 540 nM T28484 C48ADI 1190625 EC50 = 480 nM T28484 CU4PQ6 1204119 EC50 = 1800 nM T28484 C72ACT 1350845 EC50 = 5800 nM T28484 C5V1EH 2729933 IC50 = 20000 nM T28484 CTM84I 2782719 IC50 > 20000 nM T28484 CGQC14 2794294 Ki = 2659.4 nM T28484 CI6JW8 2828030 IC50 = 4300 nM T28484 C8TD6I 2849314 IC50 = 14000 nM T28484 C8J4WG 2854045 EC50 = 2600 nM T28484 CT85GW 2916332 IC50 = 1700 nM T28484 CW9O2K 2930014 IC50 = 740 nM T28484 C0T8FE 3149846 IC50 = 37200 nM T28484 CVC13H 3152075 IC50 = 5100 nM T28484 CZ02NA 3158674 IC50 = 6300 nM T28484 CK53GC 3250498 IC50 = 8500 nM T28484 C01HNZ 3333657 IC50 = 6900 nM T28484 CZ0Y4W 4252653 IC50 = 950 nM T28484 C8M6EO 4368463 IC50 = 5490 nM T28484 C0L8TM 4595895 IC50 = 15600 nM T28484 CO17EG 5015306 IC50 = 37600 nM T28484 CQ8U7S 5205832 IC50 = 40180 nM T28484 COFC26 5546231 IC50 = 134 nM T28484 CR54XC 5777336 IC50 = 4600 nM T28484 CPV72R 6102824 IC50 = 2 nM T28484 CC8W0A 6857690 IC50 = 104 nM T28484 CJZ03U 6951058 IC50 > 63000 nM T28484 CQE2S4 7009563 IC50 > 63000 nM T28484 CWV64N 7019695 IC50 > 63000 nM T28484 CQM5F8 7271796 Ki = 98.6 nM T28484 C9ZP2B 7408363 IC50 > 63000 nM T28484 CZAN92 7472794 Ki = 9.1 nM T28484 C2R8BH 9541651 IC50 = 79100 nM T28484 CSI60M 9826132 IC50 = 16 nM T28484 CLV23Q 9860103 IC50 = 9700 nM T28484 CZ2AS9 9872853 IC50 = 80 nM T28484 C5WNF7 9883349 IC50 = 450 nM T28484 COP96L 9936388 Ki = 0.5 nM T28484 CDCM57 10094631 IC50 = 23000 nM T28484 C6IVA1 10149544 IC50 = 94 nM T28484 CG1UO8 10171750 IC50 = 9800 nM T28484 CYQ3O8 10172040 IC50 = 1200 nM T28484 CH5FK7 10172108 IC50 = 1800 nM T28484 C89RTM 10193550 IC50 = 903 nM T28484 C0HA8L 10195027 IC50 = 585 nM T28484 C4X6CV 10195768 IC50 = 100 nM T28484 CFVG49 10215371 IC50 = 1100 nM T28484 CG32IU 10220615 IC50 = 18400 nM T28484 CAI34D 10236493 IC50 = 3600 nM T28484 C5LI3A 10236645 IC50 = 51 nM T28484 COM49U 10238126 IC50 = 122 nM T28484 CHGS73 10286584 IC50 = 84 nM T28484 C2L7MH 10308676 IC50 = 284 nM T28484 C61ZHJ 10309476 IC50 = 44 nM T28484 C92FJO 10309662 IC50 = 55 nM T28484 CG42HR 10310151 IC50 = 103 nM T28484 CIUH41 10357373 IC50 = 4000 nM T28484 CYA1F4 10390836 IC50 = 51 nM T28484 CIE20X 10429690 Ki = 120 nM T28484 CY9F6J 10665491 EC50 = 294 nM T28484 C1D7CQ 10968573 IC50 = 720 nM T28484 CAI5X4 10989172 IC50 > 10000 nM T28484 C80FNI 11151953 IC50 = 170 nM T28484 CYW48K 11163025 IC50 = 120 nM T28484 CN3VF5 11163393 IC50 = 110 nM T28484 C7PQ1X 11163979 IC50 = 502 nM T28484 C9NJ1E 11167161 IC50 > 63000 nM T28484 C1JZX8 11175005 IC50 = 685 nM T28484 CC60IS 11176379 IC50 = 319 nM T28484 CZD62W 11185891 IC50 = 130 nM T28484 C7D0RG 11189426 IC50 = 860 nM T28484 C8KO4G 11232296 IC50 = 6000 nM T28484 CHL4C9 11232827 IC50 = 349 nM T28484 CT18DU 11244423 IC50 = 167 nM T28484 CUS5X6 11244531 IC50 = 15 nM T28484 CJL85B 11261882 IC50 = 49 nM T28484 CAY58Q 11278857 IC50 = 120 nM T28484 C76WDK 11280370 IC50 = 67 nM T28484 C4KOJ2 11290427 IC50 = 1422 nM T28484 CE65DY 11300450 IC50 = 420 nM T28484 CSX9R5 11325207 IC50 = 40 nM T28484 C0W9YB 11336022 Ki = 110 nM T28484 CVIO67 11337670 IC50 = 39 nM T28484 C61VAJ 11348021 IC50 = 31 nM T28484 CDVR87 11348100 IC50 = 792 nM T28484 CEI5U8 11351844 IC50 = 120 nM T28484 C63JHU 11359430 IC50 = 141 nM T28484 CC3VS1 11359945 IC50 = 66 nM T28484 CX1Q6E 11382921 IC50 = 86 nM T28484 CHR14M 11392225 IC50 = 130 nM T28484 CY32TM 11393385 IC50 = 24 nM T28484 CUB4A2 11405234 IC50 = 1448 nM T28484 CH4O8V 11417613 IC50 = 176 nM T28484 CS48KQ 11427185 IC50 = 482 nM T28484 CU5XJ8 11428074 IC50 = 67 nM T28484 CKY2G7 11439836 IC50 = 28 nM T28484 CH6J7A 11450574 IC50 = 34 nM T28484 C64QZF 11461630 IC50 = 2518 nM T28484 CXR6L7 11472221 IC50 = 500 nM T28484 C58GVP 11473294 IC50 = 196 nM T28484 CU5Q4D 11473399 IC50 = 1795 nM T28484 C41CXQ 11484241 IC50 = 25 nM T28484 C5ZR9B 11492539 IC50 = 270 nM T28484 C4D6GJ 11493466 Ki = 330 nM T28484 CV41ER 11494867 IC50 = 1.8 nM T28484 C4ZLJ2 11496836 IC50 = 5 nM T28484 C1W8SH 11497413 IC50 = 4.7 nM T28484 C18KEB 11507070 IC50 = 550 nM T28484 CV4IZ7 11509189 EC50 = 3.2 nM T28484 CQEZ41 11514833 IC50 = 85 nM T28484 CTA7M3 11517739 IC50 = 4.3 nM T28484 CC19SE 11518697 IC50 = 3.9 nM T28484 C78DKQ 11539390 IC50 = 1 nM T28484 CF52ZB 11545686 IC50 = 1.6 nM T28484 CHT8D7 11547260 IC50 = 2.8 nM T28484 CL9OM0 11552755 IC50 = 2.1 nM T28484 CJ0U7Q 11577209 EC50 = 208 nM T28484 CVIP95 11582321 IC50 = 1 nM T28484 C42QMA 11590877 IC50 = 3.8 nM T28484 CM4Q2B 11597510 IC50 = 4 nM T28484 C6KVY0 11598137 IC50 = 0.9 nM T28484 C1WI4H 11611859 IC50 = 0.4 nM T28484 CD2H3T 11624832 IC50 = 5.2 nM T28484 C3M2LO 11626574 EC50 = 368 nM T28484 CV7F1O 11626838 EC50 = 27 nM T28484 CJBR83 11634073 IC50 = 1.5 nM T28484 C98YKB 11653811 IC50 = 0.2 nM T28484 CGU87J 11654962 IC50 = 1 nM T28484 CKP76R 11662966 IC50 = 1.6 nM T28484 CV62EQ 11666731 IC50 = 155 nM T28484 CMW4Y3 11668820 IC50 = 1.8 nM T28484 C29PWK 11675645 IC50 = 2.6 nM T28484 CT92YC 11680877 IC50 = 120 nM T28484 CKH1U0 11687592 IC50 > 20000 nM T28484 CWX2F0 11696319 IC50 = 0.5 nM T28484 CD0V1M 11709173 Ki = 6.8 nM T28484 CC74PN 11718862 IC50 = 1.8 nM T28484 C3FP8J 11720191 IC50 = 1 nM T28484 C70FVG 11738796 IC50 = 1100 nM T28484 CVYG50 11739086 IC50 = 2780 nM T28484 CG4Z7P 11771970 Ki = 3.5 nM T28484 CS5XA3 11772457 IC50 = 20 nM T28484 C4MJS7 11840968 IC50 = 38 nM T28484 CRSJ15 11848366 IC50 = 0.82 nM T28484 CGA83V 11853779 IC50 = 100 nM T28484 CJO8L1 11858360 IC50 = 64 nM T28484 C74LXB 11858424 IC50 = 110 nM T28484 C9YX7P 12000936 Ki = 1.4 nM T28484 CZ38QX 12984537 IC50 > 20000 nM T28484 CI30WH 13008994 Ki = 21.5 nM T28484 C0PXW1 13830550 Ki = 2157.6 nM T28484 C0YBV3 13943580 Ki = 750 nM T28484 CZ6O1D 14081820 IC50 > 63000 nM T28484 C3KP6Q 14741508 IC50 > 50000 nM T28484 C0TLA5 14855134 IC50 > 6300 nM T28484 C9ZO7G 15604796 IC50 = 1.9 nM T28484 CVKB58 15942673 IC50 = 110 nM T28484 CLD0M2 15949839 IC50 = 7 nM T28484 CUS3W4 15950258 IC50 = 7.4 nM T28484 CY09XF 15984121 IC50 = 60 nM T28484 C8F9HI 16122639 EC50 = 1700 nM T28484 C1V0YD 18686366 IC50 = 6800 nM T28484 C1QTG3 19589351 IC50 = 1900 nM T28484 CFIY91 20100158 IC50 = 1470 nM T28484 C1AFL3 21117270 Ki = 1500 nM T28484 C7FT6V 21140145 Ki < 50 nM T28484 CVZ7G3 21140146 Ki = 2000 nM T28484 CBA68L 21144445 Ki = 4.2 nM T28484 CYJ46Z 21144451 Ki = 600 nM T28484 CLJ56D 21144473 Ki = 14000 nM T28484 COXV07 22179981 IC50 = 70 nM T28484 C8X0MA 22179983 IC50 = 330 nM T28484 CXH2R9 22179996 IC50 = 60 nM T28484 CU9M1H 22180000 IC50 > 25000 nM T28484 C41IWK 22180008 IC50 = 3720 nM T28484 C0E6HG 22180029 IC50 = 100 nM T28484 CBV96L 22180034 IC50 = 1920 nM T28484 CPK6E5 22180046 IC50 = 290 nM T28484 CK7A3G 22180056 IC50 = 650 nM T28484 CM5A6D 22180071 IC50 = 60 nM T28484 C8EO1I 22185227 IC50 = 52 nM T28484 CTE52X 22577556 IC50 = 41500 nM T28484 C0RA2X 23625977 IC50 > 20000 nM T28484 C73MLP 23625981 IC50 > 20000 nM T28484 CHD2W4 23625982 IC50 = 840 nM T28484 C82PAY 23625983 IC50 > 20000 nM T28484 C3FQI4 23625984 IC50 > 20000 nM T28484 CGHE36 23626137 IC50 = 118 nM T28484 CA9JV8 23626138 IC50 > 20000 nM T28484 C8OF6I 23626140 IC50 > 20000 nM T28484 C5E7MR 23626141 IC50 > 20000 nM T28484 C32QNZ 23626142 IC50 > 20000 nM T28484 C4HC0U 23626448 IC50 = 2470 nM T28484 CY1QW4 23628220 EC50 = 100 nM T28484 C87DFY 24806224 Ki = 450 nM T28484 C80ABE 24806225 Ki < 50 nM T28484 CF9B4Q 24806226 Ki = 150 nM T28484 C25EDC 24806227 Ki = 175 nM T28484 CK8NI7 24860487 Ki = 2500 nM T28484 C1IJZ4 24860488 Ki = 4000 nM T28484 CURN19 24860489 Ki = 7000 nM T28484 CU0ZL5 24860490 Ki = 600 nM T28484 C0ADM2 24860491 Ki = 1500 nM T28484 CM52YG 24860492 Ki = 6750 nM T28484 C53JWM 24860493 Ki = 150 nM T28484 CRVG54 24860494 IC50 = 26.8 nM T28484 CEVI14 24860495 Ki = 13.6 nM T28484 CX83YD 24860496 Ki = 23000 nM T28484 CKX7A6 24860497 Ki = 35000 nM T28484 CW4SJ6 24860498 Ki = 23000 nM T28484 CAY0Z3 24860499 Ki = 1000 nM T28484 C3UT1C 24860500 Ki = 1500 nM T28484 CBA6Q2 24860501 Ki = 13000 nM T28484 C73OHZ 24860502 Ki = 6000 nM T28484 C61VPR 24860504 Ki = 900 nM T28484 CP63DU 24901489 IC50 = 85 nM T28484 C9E0OD 24901490 IC50 = 113 nM T28484 CT8GA0 24901491 IC50 = 50 nM T28484 CY3C1U 24901492 IC50 = 16 nM T28484 CC2GE7 24901493 IC50 = 5.2 nM T28484 CFM1P2 24901494 IC50 = 3.6 nM T28484 CIN21Y 24901495 IC50 = 3100 nM T28484 CF24OR 24901496 IC50 = 2.7 nM T28484 CAUZ61 24901497 IC50 = 11 nM T28484 C7IQO2 24901498 IC50 = 24.7 nM T28484 C8QOY5 24901499 IC50 = 3140 nM T28484 C93PNA 24901500 IC50 = 606 nM T28484 CBG32M 24901501 IC50 = 745 nM T28484 C2E1YR 24901502 IC50 = 697 nM T28484 CC54GX 24901503 IC50 = 390 nM T28484 CA0R5M 24901504 IC50 = 67 nM T28484 C07IFO 24901505 IC50 = 119 nM T28484 CANF39 24901506 IC50 = 892 nM T28484 CY38XS 24901507 IC50 = 391 nM T28484 CMC52T 24901508 IC50 = 552 nM T28484 C0XHP1 24901509 IC50 = 686 nM T28484 CS3W4I 24901510 IC50 = 8 nM T28484 CBV2S9 24901511 IC50 = 26 nM T28484 CN2K8P 24901512 IC50 = 85 nM T28484 CX5TH2 24901513 IC50 = 4 nM T28484 C6YGU7 24901514 IC50 = 16.5 nM T28484 CY3EB5 24901515 EC50 = 53 nM T28484 CTHL35 24901516 IC50 = 5.2 nM T28484 C1V3QA 24901517 IC50 = 3.8 nM T28484 COCN23 24901519 IC50 = 8230 nM T28484 CJ8LU2 24901520 IC50 = 25200 nM T28484 CBGF57 24901521 IC50 = 11000 nM T28484 CY1CW5 24901522 IC50 > 25000 nM T28484 CML92E 24901523 IC50 = 2270 nM T28484 CAM5I2 24901524 IC50 = 3060 nM T28484 CK1UJ2 24901525 IC50 = 4650 nM T28484 CO1Z9X 24901526 IC50 > 25000 nM T28484 C3QHP5 24901527 IC50 = 8880 nM T28484 CDYR21 24901528 IC50 = 5360 nM T28484 CQXW01 24901529 IC50 = 17900 nM T28484 CJK3F0 24901530 IC50 = 16400 nM T28484 CCHV96 24901531 IC50 > 25000 nM T28484 CV59OA 24901532 IC50 = 14400 nM T28484 CH0J7C 24901533 IC50 > 25000 nM T28484 C7J3LO 24901534 IC50 > 25000 nM T28484 CY05BM 24901535 IC50 > 25000 nM T28484 C3KUV2 24901536 IC50 = 2750 nM T28484 CZ04WL 24901537 IC50 = 22300 nM T28484 CTY2R8 24901538 IC50 = 12800 nM T28484 C5V6ZS 24901539 IC50 = 5440 nM T28484 C7QOX2 24901540 IC50 = 306 nM T28484 C3EDI4 24901541 IC50 > 25000 nM T28484 CT6N0Z 24901542 IC50 = 13200 nM T28484 C4D2NY 24901543 IC50 = 3480 nM T28484 CY0P8H 24901544 IC50 > 25000 nM T28484 C5WQ9S 24901545 IC50 > 25000 nM T28484 C3RY1T 24901546 IC50 = 2490 nM T28484 CE56RM 24901547 IC50 = 808 nM T28484 C9AL2E 24901548 IC50 = 317 nM T28484 C79OHQ 24901549 IC50 = 595 nM T28484 CF14PC 24901550 IC50 = 617 nM T28484 C7N0YQ 24901551 IC50 > 25000 nM T28484 CT4G9C 24901552 IC50 > 25000 nM T28484 C97OEW 24901553 IC50 > 25000 nM T28484 C58DLP 24901554 IC50 = 4710 nM T28484 CY5TL9 24901555 IC50 = 344 nM T28484 CCBU08 24901556 IC50 = 1780 nM T28484 C5R6AJ 24901557 IC50 = 12800 nM T28484 CR61YE 24901558 IC50 = 1270 nM T28484 C1FPG9 24901560 IC50 = 639 nM T28484 C8T5CB 24901561 EC50 < 30000 nM T28484 CT1H2D 24901562 EC50 = 29000 nM T28484 C1D4VU 24901563 EC50 = 4300 nM T28484 C1C8HQ 24901564 IC50 = 76000 nM T28484 CG0O1W 24901565 IC50 = 17000 nM T28484 C7SFY5 24901567 EC50 = 1100 nM T28484 C15JND 24901568 EC50 = 37000 nM T28484 CSGI87 24901569 EC50 = 7600 nM T28484 CE43VJ 24901570 EC50 = 4700 nM T28484 COPT12 24901571 EC50 = 5400 nM T28484 C13QJL 24901572 EC50 = 1500 nM T28484 CP7C8W 24901573 IC50 = 12000 nM T28484 CBN3V7 24901574 EC50 = 1900 nM T28484 C8IC1E 24901575 IC50 = 69000 nM T28484 C10ZYD 24901576 EC50 = 17000 nM T28484 C9QA1U 24901577 IC50 = 3300 nM T28484 CH4T2K 24901578 EC50 < 30000 nM T28484 CXO6N4 24901579 EC50 < 30000 nM T28484 C5BL4Q 25014675 IC50 = 14800 nM T28484 C69ZRO 25014747 Ki < 50 nM T28484 COX3F5 25014748 IC50 = 514.2 nM T28484 CCI29G 25014750 IC50 = 680 nM T28484 CAW3B7 25014751 IC50 > 63000 nM T28484 C53QJP 25015247 IC50 = 230 nM T28484 CPLY38 25164463 IC50 > 20000 nM T28484 CAXQ03 25164661 IC50 = 7400 nM T28484 CRU76E 25164662 IC50 > 20000 nM T28484 C3NVW5 25165471 IC50 = 2500 nM T28484 CV6Y1Z 25165472 IC50 = 5000 nM T28484 CVMZ57 25165473 IC50 = 6900 nM T28484 CF9KY4 25165474 IC50 = 4800 nM T28484 CIWL28 25165475 IC50 = 1400 nM T28484 CPV3O6 25165666 IC50 = 458.8 nM T28484 C56QHJ 25165854 IC50 = 1300 nM T28484 C37LFS 25166248 IC50 = 7900 nM T28484 C25CJK 25184242 IC50 = 420 nM T28484 CB9H1A 25184517 IC50 = 1400 nM T28484 CCA5X7 25184518 IC50 = 7140 nM T28484 CQG3B5 25184521 IC50 = 1470 nM T28484 CT17QC 25184589 IC50 = 3630 nM T28484 C76VQM 25184659 IC50 = 3700 nM T28484 C3U5KV 25229667 EC50 = 139 nM T28484 CK1DA7 26367385 IC50 > 10000 nM T28484 CL60OC 26367815 IC50 > 10000 nM T28484 CWI2E1 29066543 IC50 > 6300 nM T28484 C1IGM6 42633262 EC50 = 3313 nM T28484 CT9V6K 42633458 EC50 = 246 nM T28484 CURL76 42633808 EC50 > 1000 nM T28484 CFUL48 42633810 EC50 > 1000 nM T28484 CW53FJ 42634875 EC50 > 1000 nM T28484 CE1VH8 42634877 EC50 > 500 nM T28484 CFY4X2 42634878 EC50 = 338 nM T28484 CSYR62 42635606 EC50 = 452 nM T28484 C83DTG 42635776 EC50 = 665 nM T28484 CD86FT 43132780 IC50 > 6300 nM T28484 C2TA6X 44130714 IC50 = 20 nM T28484 C5HA7I 44130820 IC50 = 40 nM T28484 CSVI35 44130821 IC50 = 60 nM T28484 CH58RQ 44187469 IC50 = 40 nM T28484 CY8UD3 44238920 IC50 = 46200 nM T28484 C0R8XE 44401424 IC50 > 5000 nM T28484 CK19QO 44401630 IC50 = 460 nM T28484 C8AE7V 44401700 IC50 = 23300 nM T28484 CH5NI0 44401702 IC50 = 10900 nM T28484 CD5GA9 44401759 IC50 = 13500 nM T28484 CA3Z6Q 44401762 IC50 = 250 nM T28484 CEM2V4 44401802 IC50 = 1800 nM T28484 CYZ40J 44401803 IC50 = 3600 nM T28484 CO8U3T 44401822 IC50 = 12700 nM T28484 CXN82K 44401861 IC50 = 6000 nM T28484 CLR2J1 44401864 IC50 > 50000 nM T28484 C53MQP 44401865 IC50 > 50000 nM T28484 COL4M1 44401990 IC50 > 50000 nM T28484 C6TZW3 44401991 IC50 > 50000 nM T28484 CH9L1R 44409515 IC50 = 50000 nM T28484 CB91NT 44409718 IC50 = 13 nM T28484 C5YP1R 44409879 IC50 = 1.3 nM T28484 CKI20Y 44409884 IC50 = 4 nM T28484 C39MWE 44409885 IC50 = 5.5 nM T28484 CF8A0Z 44409903 IC50 = 1.2 nM T28484 CYO7B5 44409904 IC50 = 0.5 nM T28484 C7BM2G 44409905 IC50 = 2.9 nM T28484 C2W8UD 44414670 IC50 = 980 nM T28484 CZX6L4 44414697 IC50 = 190 nM T28484 CET0G6 44414850 IC50 = 6880 nM T28484 CS76CV 44414851 IC50 = 6060 nM T28484 CK16MO 44426727 IC50 = 20000 nM T28484 CZ6RH3 44426731 IC50 = 26 nM T28484 CON04H 44430571 IC50 = 2.2 nM T28484 C7L0PH 44430573 IC50 = 10.2 nM T28484 CDA0X6 44430574 IC50 = 10.2 nM T28484 CT6HC8 44430575 IC50 = 12.1 nM T28484 C7LQ2E 44430576 IC50 = 110 nM T28484 CCBR69 44430578 IC50 = 5.2 nM T28484 CFW02R 44432703 IC50 = 3100 nM T28484 CG78BW 44435327 IC50 = 5000 nM T28484 CSY1J0 44435339 IC50 = 3800 nM T28484 CVS9Y7 44435350 IC50 = 0.9 nM T28484 C74VGT 44435351 IC50 = 1.4 nM T28484 C1FK4E 44435373 IC50 = 1 nM T28484 CXW8Q9 44435374 IC50 = 1.3 nM T28484 CPMN93 44435375 IC50 = 1 nM T28484 CD4EI7 44435376 IC50 = 2 nM T28484 CEX75D 44435377 IC50 = 5.2 nM T28484 COX3Q2 44442283 IC50 = 1.8 nM T28484 C2DZI3 44442301 IC50 = 3 nM T28484 C53HAL 44442302 IC50 = 800 nM T28484 CKJ0Y7 44442887 IC50 = 1.2 nM T28484 CDR7O2 44444939 IC50 = 6600 nM T28484 C4X5PE 44444940 IC50 = 15000 nM T28484 CCL96S 44444941 IC50 = 27000 nM T28484 C6LVI5 44445386 IC50 = 12 nM T28484 CL6YR4 44445387 IC50 = 280 nM T28484 CA82IF 44576259 IC50 = 150 nM T28484 C0JO7X 44590391 IC50 > 20000 nM T28484 CR68ES 44590392 IC50 = 2140 nM T28484 C79YFQ 44590435 IC50 > 20000 nM T28484 CXQE68 44590436 IC50 > 20000 nM T28484 C8O9MZ 44590437 IC50 = 120 nM T28484 CH1S4F 44590510 IC50 = 4610 nM T28484 CMDR03 44590511 IC50 > 20000 nM T28484 CA37FS 44590512 IC50 = 860 nM T28484 CQ1SU4 44590513 IC50 > 20000 nM T28484 COK1F0 44590548 IC50 = 3060 nM T28484 CAG9D7 44590549 IC50 = 700 nM T28484 C1FCO0 45266928 IC50 = 6000 nM T28484 C1Y4KO 45267020 IC50 > 20000 nM T28484 CLK10E 45267851 IC50 = 19000 nM T28484 C53DIE 45267853 IC50 = 520 nM T28484 CO5BT3 45267860 IC50 = 5200 nM T28484 C93RCK 45267863 IC50 > 20000 nM T28484 CAWS46 45267869 IC50 > 20000 nM T28484 C0C7UM 45267870 IC50 > 20000 nM T28484 CK60GY 45267896 IC50 > 20000 nM T28484 C71NGE 45268737 IC50 = 9200 nM T28484 C2ZN5S 45268741 IC50 > 20000 nM T28484 CP4M3X 45268781 IC50 = 20000 nM T28484 C9GJA6 45269595 IC50 = 16300 nM T28484 CTW13H 45269596 IC50 > 20000 nM T28484 C96UFG 45270431 IC50 = 13400 nM T28484 CZ5ID2 45271261 IC50 = 2400 nM T28484 C0X5FN 45271263 IC50 > 20000 nM T28484 CER7W9 45271267 IC50 > 50000 nM T28484 C32JIV 45271285 IC50 > 20000 nM T28484 CN32MP 45272152 IC50 = 33400 nM T28484 CATM09 45272155 IC50 > 20000 nM T28484 C8SB6M 45272157 IC50 > 20000 nM T28484 C70MZU 45272180 IC50 > 20000 nM T28484 C3SRC5 45272183 IC50 > 20000 nM T28484 CRT26A 45272991 IC50 = 2100 nM T28484 CG9XA3 45272994 IC50 = 2200 nM T28484 C3P2WK 45272999 IC50 > 20000 nM T28484 CRUZ63 45789422 IC50 = 20 nM T28484 CRK61L 46224756 IC50 = 155 nM T28484 C7U0NT 46224757 IC50 = 760 nM T28484 CR09DX 46224758 IC50 = 8100 nM T28484 C9DA2G 46224759 IC50 = 175 nM T28484 CC1K2T 46224798 IC50 = 11000 nM T28484 C1SW2H 46224799 IC50 > 25000 nM T28484 C5R3XW 46224800 IC50 > 25000 nM T28484 CBE70W 46224801 IC50 > 25000 nM T28484 C0F6LC 46224802 IC50 = 6600 nM T28484 CI0EG3 46224838 IC50 = 230 nM T28484 CA87WH 46224839 IC50 = 100 nM T28484 CD2ZR7 46224840 IC50 = 200 nM T28484 CGN91R 46225130 IC50 = 630 nM T28484 C59QCL 46225171 IC50 = 760 nM T28484 CVM2D6 46225172 IC50 = 11 nM T28484 C5ZTB8 46225173 IC50 > 25000 nM T28484 C1G8XD 46225174 IC50 = 1700 nM T28484 CF87SZ 46225213 IC50 = 27 nM T28484 C8RSW5 46225214 IC50 = 4500 nM T28484 CWR71G 46225215 IC50 = 200 nM T28484 CW8E2J 46225216 IC50 = 460 nM T28484 CLHF47 46225271 IC50 = 49 nM T28484 CW7H9X 46225272 IC50 = 186 nM T28484 CBC20V 46225273 IC50 = 100 nM T28484 CB3L9I 46225274 IC50 = 900 nM T28484 C3AXM5 46244083 IC50 > 6300 nM T28484 CZ93BW 46244085 IC50 = 95 nM T28484 CWLZ72 46244164 IC50 = 31 nM T28484 C9BGT3 46244165 IC50 = 84 nM T28484 CRZ2Y8 46881445 IC50 = 300 nM T28484 CPZH92 46881446 IC50 > 10000 nM T28484 C38PRQ 46881447 IC50 = 530 nM T28484 CXUQ18 46881495 IC50 > 10000 nM T28484 CFH1G2 46881496 IC50 > 10000 nM T28484 C87UKL 46881497 IC50 = 11 nM T28484 C4SN5I 46881539 IC50 = 14 nM T28484 CGRJ18 46881540 IC50 = 4 nM T28484 C0K3ZJ 46881541 IC50 = 7 nM T28484 CG4W0M 46881581 IC50 = 19 nM T28484 C5SR9E 46881582 IC50 = 65 nM T28484 CL37QK 46881583 IC50 = 6 nM T28484 CVG3U7 46881584 IC50 = 4 nM T28484 C5BLY4 46881627 IC50 = 58 nM T28484 C0T2QG 46881628 IC50 = 4 nM T28484 CIOR36 46881629 IC50 = 19 nM T28484 CK69QD 46881630 IC50 = 5 nM T28484 CWH96P 46881663 IC50 = 11 nM T28484 CDXM14 46881664 IC50 = 2 nM T28484 C3N7QJ 46881665 IC50 = 3 nM T28484 COJ2Z3 46881666 IC50 = 6 nM T28484 CV51NZ 46881710 IC50 = 5 nM T28484 C10HXD 46881711 IC50 = 7 nM T28484 CZ0BX5 46881712 IC50 = 2 nM T28484 CH70VR 46881713 IC50 > 10000 nM T28484 CRZ4S6 46881714 IC50 = 300 nM T28484 C38SKH 46881763 IC50 = 870 nM T28484 CS0QT5 46881764 IC50 = 10000 nM T28484 C5WA2J 46881841 IC50 = 360 nM T28484 CL25ZI 46881873 IC50 = 910 nM T28484 CAX5T3 46881905 IC50 = 3700 nM T28484 CA2S0Z 46881906 IC50 > 10000 nM T28484 C7TS6M 46881907 IC50 = 5300 nM T28484 C9AB2L 46881943 IC50 = 10000 nM T28484 CP4K8C 46881944 IC50 > 10000 nM T28484 CR2J7M 46881945 IC50 = 90 nM T28484 C4QPY2 46881946 IC50 = 540 nM T28484 C8ZJ0N 46881947 IC50 = 1250 nM T28484 CJ3QP9 46881992 IC50 > 10000 nM T28484 C5O7KT 46881993 IC50 = 95 nM T28484 CKY96D 46882035 IC50 = 17 nM T28484 C7OZ6P 46882036 IC50 > 10000 nM T28484 C40WET 46882037 IC50 > 10000 nM T28484 CAI32G 46882038 IC50 = 2300 nM T28484 CKA9Z2 46882039 IC50 > 10000 nM T28484 CA56YD 46882089 IC50 = 270 nM T28484 CUN64R 46882090 IC50 = 350 nM T28484 C3Y7CF 46882091 IC50 = 6800 nM T28484 CN74LO 46906141 IC50 = 724 nM T28484 CYE46T 46906142 IC50 = 75 nM T28484 C3DP7L 46906178 IC50 = 224 nM T28484 CU0LO3 46906179 IC50 = 380 nM T28484 CW75MT 46906180 IC50 = 118 nM T28484 C6W0RZ 46906181 IC50 = 3453 nM T28484 CTD9Y2 46906182 IC50 = 290 nM T28484 CN35PL 46906232 IC50 = 65 nM T28484 CEC3U2 46906234 IC50 = 483 nM T28484 C1DE9K 46906236 IC50 = 40 nM T28484 CI31VX 46906237 IC50 = 76 nM T28484 CK0X7D 46906238 IC50 = 50 nM T28484 C45BIP 46906260 IC50 = 664 nM T28484 C52VRS 46906261 IC50 = 169 nM T28484 CVWR15 46906262 IC50 = 710 nM T28484 C1CW4B 46906263 IC50 = 462 nM T28484 CG75KB 46906264 IC50 = 12378 nM T28484 CKI5A6 46906288 IC50 = 237 nM T28484 CFM5E4 46906290 IC50 = 83 nM T28484 C5RJ2A 46906292 IC50 = 454 nM T28484 CYT0O2 46906294 IC50 = 7 nM T28484 C3WFU8 46906296 IC50 = 204 nM T28484 C42KOP 46906327 IC50 = 347 nM T28484 CKLA96 46906328 IC50 = 51 nM T28484 CEI4X2 46906329 IC50 = 216 nM T28484 CV95BH 46906358 IC50 < 1 nM T28484 CW1H5I 46906359 IC50 = 337 nM T28484 C7OJD1 46906360 IC50 = 1703 nM T28484 CB47DW 46906361 IC50 = 163 nM T28484 C0QEB1 46906363 IC50 = 43 nM T28484 CX87SF 49772558 IC50 = 800 nM T28484 CW3A2L 50901410 EC50 = 1 nM T28484 CY89XM 51356550 IC50 = 1578 nM T28484 C1I7YM 51356551 Ki = 1349.7 nM T28484 C9G6RQ 51356552 Ki = 428.6 nM T28484 C46KAO 51356553 Ki = 84.2 nM T28484 C5AFN6 51356813 Ki < 50 nM T28484 C6N2LD 51356814 Ki < 50 nM T28484 CO6Y8P 51356815 Ki < 50 nM T28484 CU3V9I 51356816 IC50 = 21.8 nM T28484 CR23LH 51356817 IC50 = 19.3 nM T28484 CMCX63 51356818 Ki = 76.2 nM T28484 C1SB5L 51356819 Ki = 302.1 nM T28484 CJU3O1 53326599 IC50 = 41700 nM T28484 C0XG9J 53363371 IC50 = 37 nM T28484 C7HB2V 53363372 IC50 = 45 nM T28484 CQ0S7J 53363455 IC50 = 170 nM T28484 C5BDJ3 53363538 IC50 = 330 nM T28484 CO8AN7 53363539 IC50 = 40 nM T28484 CQ70WO 53363540 IC50 = 180 nM T28484 C45PEV 53363541 IC50 = 58 nM T28484 CN65FT 53363542 IC50 = 45 nM T28484 CTZ1V6 53494967 IC50 = 11 nM T28484 CDI45K 53494981 EC50 = 190 nM T28484 CUQ57S 54757107 IC50 = 10 nM T28484 CMU2H3 54757108 IC50 = 140 nM T28484 C4HTS9 54757109 IC50 = 20 nM T28484 CYMF79 54757209 IC50 = 210 nM T28484 C5LK6A 54757210 IC50 = 130 nM T28484 C6ATD7 54757211 IC50 = 160 nM T28484 CWF67S 54757212 IC50 = 760 nM T28484 CZTJ96 54757416 IC50 = 3500 nM T28484 CDF4W5 54757520 IC50 = 3800 nM T28484 C7MY9B 54757521 IC50 = 5310 nM T28484 CVLZ09 54757522 IC50 = 630 nM T28484 CSX2J4 54757523 IC50 = 9090 nM T28484 C0JZP8 54757524 IC50 = 9000 nM T28484 CSH5W0 54757525 IC50 = 390 nM T28484 CSXE03 54757628 IC50 = 310 nM T28484 CP05UA 54757629 IC50 = 1070 nM T28484 C4JNP8 54757630 IC50 = 1440 nM T28484 CI4K2Y 54757631 IC50 = 2920 nM T28484 CGA3F2 54757632 IC50 = 5990 nM T28484 C4ANQ9 54757740 IC50 = 10000 nM T28484 C76OHM 54757741 IC50 = 5520 nM T28484 CU67QC 54757742 IC50 = 4540 nM T28484 CAY9J2 54757743 IC50 = 6700 nM T28484 C6MG0Y 54757744 IC50 = 4220 nM T28484 CXG51Q 54757745 IC50 = 9000 nM T28484 C9YSJ5 54757838 IC50 = 200 nM T28484 CG41NO 54757839 IC50 = 610 nM T28484 CDE51C 54757840 IC50 = 50 nM T28484 C16YBT 54757841 IC50 = 150 nM T28484 CJV92T 54757842 IC50 = 30 nM T28484 CSQ18G 54757932 IC50 = 210 nM T28484 C1OPZ7 54757933 IC50 = 310 nM T28484 C1UGW3 54757934 IC50 = 2460 nM T28484 C9VO5E 54757935 IC50 = 90 nM T28484 CP39EO 54757936 IC50 = 1060 nM T28484 CGPF63 54758031 IC50 = 20 nM T28484 CL81AQ 54758032 IC50 = 90 nM T28484 CHK86M 54758034 IC50 = 940 nM T28484 C2G6FN 54758035 IC50 = 210 nM T28484 C50VBJ 54758036 IC50 = 140 nM T28484 CE7UF4 54758123 IC50 = 2700 nM T28484 C5KXB9 54758124 IC50 = 5960 nM T28484 CZV8K4 54758125 IC50 = 500 nM T28484 C43ZMD 54758126 IC50 = 1390 nM T28484 CKTN03 54758127 IC50 = 410 nM T28484 C8S0LO 54758216 IC50 = 980 nM T28484 CN4HU9 54758217 IC50 = 2310 nM T28484 CUW4I9 54758219 IC50 = 40 nM T28484 CGZ87Q 54758220 IC50 = 3210 nM T28484 CLF81J 54758305 IC50 = 30 nM T28484 C1RL6Q 54758306 IC50 = 150 nM T28484 C1I7AT 54758307 IC50 = 13 nM T28484 CJZ7W0 54758308 IC50 = 21 nM T28484 CI30OS 54758309 IC50 = 1900 nM T28484 CZHK43 54758400 IC50 = 141 nM T28484 C80NZC 54758401 IC50 = 85 nM T28484 C78BQR 54758402 IC50 = 161 nM T28484 CB1WF5 54758404 IC50 = 323 nM T28484 CSEO14 54758405 IC50 = 5460 nM T28484 CDCG23 54763606 IC50 = 40 nM T28484 C2A5YK 56659866 IC50 = 3959 nM T28484 CVOE09 56659867 IC50 = 1047 nM T28484 CT3U4V 56659868 IC50 = 33 nM T28484 CJ64NA 56659895 IC50 = 334 nM T28484 CG05CX 56662634 EC50 = 160 nM T28484 C3QSP7 56663328 IC50 = 146 nM T28484 CQV76H 56663329 IC50 = 169 nM T28484 COQ9D7 56663330 IC50 = 73 nM T28484 C5UMQ0 56666752 IC50 = 2345 nM T28484 C3G5ZI 56666753 IC50 = 1307 nM T28484 C0VMD1 56670186 IC50 = 232 nM T28484 CYI76G 56670187 IC50 = 1485 nM T28484 CWY2M5 56670188 IC50 = 20 nM T28484 CNTE86 56670189 IC50 = 42 nM T28484 CFH4K0 56670190 IC50 = 9925 nM T28484 CCN9I5 56670191 IC50 = 92 nM T28484 CBU09F 56673708 IC50 = 3409 nM T28484 CBOA18 56673709 IC50 = 49 nM T28484 CON3Y6 56673710 IC50 = 25 nM T28484 C4YLM0 56673740 IC50 = 360 nM T28484 CRJ3T6 56677019 IC50 = 1443 nM T28484 CV34UO 56677053 IC50 = 51 nM T28484 CDXF18 56680345 IC50 = 162 nM T28484 CO72KD 56680346 IC50 = 37130 nM T28484 C1NG8Y 56680347 IC50 = 2942 nM T28484 C0QYH3 56683673 IC50 = 1943 nM T28484 CO8VL4 56683674 IC50 = 828 nM T28484 C08HWQ 56683675 IC50 = 23 nM T28484 C37TXD 56683676 IC50 = 170 nM T28484 C02AUW 56683677 IC50 = 149 nM T28484 CY4KM5 56683678 IC50 = 2767 nM T28484 CTHB21 56683713 IC50 = 1178 nM T28484 CIL79O 56931000 Ki = 5.1 nM T28484 CKN0Z8 56964577 Ki = 6.4 nM T28484 CVC4F5 57325586 Ki = 173.5 nM T28484 C3LVB8 57325587 Ki = 384.4 nM T28484 CZ97DS 57325588 Ki = 3.4 nM T28484 CT67IO 57325589 Ki = 11.1 nM T28484 CO65CE 57325590 Ki = 16.7 nM T28484 C2G9UJ 57326381 Ki = 3018.5 nM T28484 CHM19P 57326382 Ki = 235.4 nM T28484 C43JBM 57326383 Ki = 1783.9 nM T28484 CC0K7O 57326384 Ki = 377.4 nM T28484 CVL16W 57326474 Ki = 89.9 nM T28484 C1K8UN 57326475 Ki = 297.8 nM T28484 C5KRE2 57326476 Ki = 293.9 nM T28484 CJF94R 57326477 Ki = 80 nM T28484 CA2C3V 57326478 Ki = 5.9 nM T28484 CG7Q0Z 57326479 Ki = 10.3 nM T28484 C6O2VB 57326480 Ki = 29.6 nM T28484 C79WOY 57326575 Ki = 352.7 nM T28484 CY04HP 57326576 Ki = 149.8 nM T28484 CAMQ75 57326577 Ki = 520.4 nM T28484 C26DYS 57326578 Ki = 27.8 nM T28484 CY5M7J 57326579 Ki = 519.8 nM T28484 CJ1XC9 57326580 Ki = 185.8 nM T28484 CA35GO 57326581 Ki = 271.7 nM T28484 CN2Q7U 57326676 Ki = 51 nM T28484 CPZG76 57326677 Ki = 120.6 nM T28484 CV5CP4 57326678 Ki = 8.8 nM T28484 CJW83U 57326679 Ki = 10.7 nM T28484 CRGX38 57326680 Ki = 7.5 nM T28484 C1O9PY 57326681 Ki = 9.7 nM T28484 C9UAK0 57326682 Ki = 1978.5 nM T28484 C6OVF0 57326778 Ki = 48.8 nM T28484 C3QI6O 57326779 Ki = 200.3 nM T28484 C93LBU 57326780 Ki = 450.6 nM T28484 C82GXC 57326781 Ki = 838.2 nM T28484 CLIY16 57326782 Ki = 829.2 nM T28484 CVG8I7 57326783 Ki = 990.6 nM T28484 C5PE0A 57326784 Ki = 329.9 nM T28484 CFER23 57326878 Ki = 419.7 nM T28484 C4QGS0 57326879 Ki = 887.8 nM T28484 C1W5BJ 57326880 Ki = 6055.6 nM T28484 CSHD25 57326881 Ki = 2089.6 nM T28484 CQ5IL7 57326882 Ki = 432.4 nM T28484 CDZ41W 57326883 Ki = 311.2 nM T28484 CI6X8L 57326884 Ki = 2942.4 nM T28484 CO12LV 57326973 Ki = 1721.3 nM T28484 CC6LV4 57326974 Ki = 3228.6 nM T28484 CSC21A 57326975 Ki = 2030.8 nM T28484 C5NSW2 57326976 Ki = 1526.7 nM T28484 CD2I1C 57326977 Ki = 1212.1 nM T28484 CVX8P7 57380650 Ki = 57.5 nM T28484 C36MNJ 57380880 Ki = 27.4 nM T28484 C9R5IA 57401215 IC50 = 1520 nM T28484 C1SYP6 57770895 IC50 = 43 nM T28484 C30GOZ 58274571 EC50 > 1000 nM T28484 CP5W0V 58274609 EC50 = 17 nM T28484 C7QN5G 58274649 EC50 = 367 nM T28484 CC9E2T 58274650 EC50 = 2 nM T28484 C0I8ZH 58274695 EC50 = 3 nM T28484 C2MVQ1 58274709 EC50 = 263 nM T28484 CEG26H 58274714 EC50 = 205 nM T28484 CRS37Y 58274722 EC50 > 1000 nM T28484 C7KF5J 58274841 EC50 = 11 nM T28484 C2CG0V 58274853 EC50 = 5 nM T28484 CM90LF 58274857 EC50 = 5 nM T28484 C8ABU3 58274876 EC50 = 179 nM T28484 CCV19B 58274954 EC50 = 615 nM T28484 CCD3W8 58274960 EC50 > 1000 nM T28484 C5C6DO 58274962 EC50 > 500 nM T28484 CC8O4I 66572223 IC50 = 15836 nM T28484 CL2F4E 66572224 IC50 > 150000 nM T28484 CA51QV 66572225 IC50 = 942.2 nM T28484 C30DFU 66572226 IC50 > 50000 nM T28484 CTU1R0 66572322 IC50 = 138 nM T28484 CM94VH 66572323 IC50 = 216.8 nM T28484 CHL76C 66572324 IC50 = 128.9 nM T28484 CCKA14 66572325 IC50 = 67.6 nM T28484 CV8W5P 66572326 IC50 = 150.5 nM T28484 CCY59V 66572327 IC50 = 58.6 nM T28484 C01MQK 66572328 IC50 = 167.6 nM T28484 CN52JC 66572329 IC50 = 159.4 nM T28484 C9KR7P 66572330 IC50 = 191.2 nM T28484 CEA8H0 66572331 IC50 = 567.5 nM T28484 CJS1P6 66572332 IC50 = 178.2 nM T28484 CO02JB 66572333 IC50 = 251.8 nM T28484 CSY2M1 66572334 IC50 = 106.5 nM T28484 CD1K4R 66572336 IC50 = 684.5 nM T28484 CA0T1V 66572337 IC50 = 789.5 nM T28484 CMDK30 66572339 IC50 = 519 nM T28484 CY4GT7 66572340 IC50 = 256.1 nM T28484 C5P8YR 66572341 IC50 = 577.9 nM T28484 CB79JX 66572342 IC50 = 140.9 nM T28484 C3PI0K 66572343 IC50 = 171.9 nM T28484 CMLZ63 66572344 IC50 = 665.6 nM T28484 C5V4JE 66572345 IC50 = 229.3 nM T28484 CZ0P4L 66572346 IC50 = 436.7 nM T28484 CP2V9F 66572347 IC50 = 587.8 nM T28484 CX2HN0 66572348 IC50 = 403.7 nM T28484 CEB16H 66572349 IC50 = 261 nM T28484 CAE28S 66572426 IC50 = 237.5 nM T28484 CX0RP9 66572427 IC50 = 455.8 nM T28484 CO0WK1 66572428 IC50 = 5278 nM T28484 CON57P 70052856 IC50 = 209 nM T28484 C02WNA 70053909 IC50 = 14 nM T28484 C37EFB 71582936 Ki = 17.3 nM T28484 C83PHC 71582937 Ki = 6.4 nM T28484 CLK98I 71582938 Ki = 6.7 nM T28484 CJ93HQ 71582939 Ki = 9.7 nM T28484 C3VKE2 71583032 Ki = 9 nM T28484 CHEZ52 71583033 Ki = 10.1 nM T28484 C5OZ9A 71583034 Ki = 128.6 nM T28484 CNUV80 71583035 Ki = 1.2 nM T28484 CJ87LP 71583036 Ki = 25.7 nM T28484 CD0K5I 71583037 Ki = 4.6 nM T28484 CKT07A 71583038 Ki = 7.8 nM T28484 CTU98Z 71583147 Ki = 2.1 nM T28484 CWO2B0 71583148 Ki = 10.6 nM T28484 CAQR82 71583149 Ki = 9.9 nM T28484 CS3W2I 71716295 Ki = 6.8 nM T28484 C8I6YH 71716296 Ki = 2268 nM T28484 C17ZJR 71716894 Ki = 4.8 nM T28484 CO3JW5 71716895 Ki = 7.8 nM T28484 CM5OR8 71716896 Ki = 27.3 nM T28484 CWGK81 71717524 Ki = 55.6 nM T28484 C1Q8JS 71718135 Ki = 201.3 nM T28484 C5F4AH 71718730 Ki = 33.6 nM T28484 CKV3Q0 71719339 Ki = 293.6 nM T28484 CHO97G 71719340 Ki = 10.1 nM T28484 CN9HI3 71719341 Ki = 162.2 nM T28484 C7CSF4 71719342 Ki = 29.7 nM T28484 C7EBW0 71719940 Ki = 11.6 nM T28484 CD3H0E 71719941 Ki = 35.2 nM T28484 C52WMG 71719942 Ki = 31.4 nM T28484 C1SHK7 71719943 Ki = 56 nM T28484 C46ATF 71720565 Ki = 37.9 nM T28484 C7OV0J 71720566 Ki = 200.3 nM T28484 C8T4SO 71720567 Ki = 64.2 nM T28484 CR5P1H 71720568 Ki = 88.4 nM T28484 C3WQ9R 71726419 IC50 = 7800 nM T28484 C1T3XH 71748071 IC50 = 75 nM T28484 CTA0Q7 71748279 IC50 = 11 nM T28484 CAU9T7 71748280 IC50 = 21 nM T28484 CT97BV 71748288 IC50 = 9.3 nM T28484 CI46YR 71748289 IC50 = 14 nM T28484 CJY8M1 71748290 IC50 = 301 nM T28484 CMSK27 71748293 IC50 = 61 nM T28484 CK6UI7 76309865 IC50 = 78 nM T28484 C7JPK0 76313576 IC50 = 123 nM T28484 C9Y6OA 76313577 IC50 = 98 nM T28484 C5DQI1 76313578 IC50 = 59 nM T28484 C9BGM3 76320800 IC50 = 67 nM T28484 CX1M2W 76320801 IC50 = 63 nM T28484 CEPO93 76324458 IC50 = 122 nM T28484 C0P1JY 76324459 IC50 = 23 nM T28484 C13EZQ 76324460 IC50 = 91 nM T28484 C6N8DX 76324461 IC50 = 168 nM T28484 CLH7P8 76324462 IC50 = 157 nM T28484 C9U0BW 76328015 IC50 = 52 nM T28484 CJ98YI 76331674 IC50 = 38 nM T28484 C2TP4I 76331675 IC50 = 170 nM T28484 CVWS93 76331676 IC50 = 76 nM T28484 C27RMF 76335284 IC50 = 27 nM T28484 CF7U1J 76335285 IC50 = 149 nM T28484 CCQ8W2 76751913 EC50 = 5 nM T28484 CZ5K3S 78319352 IC50 = 16500 nM T28484 CJAM82 82537489 IC50 = 7000 nM T28484 CMY36J 86291007 IC50 = 50 nM T28484 CP1K4E 86298441 IC50 = 35 nM T28484 C7HZS1 86342357 IC50 = 2000 nM T28484 CBGD01 86342358 IC50 = 330 nM T28484 CQ98RK 86342359 IC50 = 810 nM T28484 CQPS98 86342360 IC50 = 430 nM T28484 CUI63O 86342362 IC50 = 1200 nM T28484 CKX3I5 86342363 IC50 = 440 nM T28484 C7BDZ0 86342395 IC50 = 290 nM T28484 CM7DQ4 86342396 IC50 = 810 nM T28484 CWB36G 86342397 IC50 = 190 nM T28484 CXBK16 86342398 IC50 > 6300 nM T28484 CHQ4L6 86342400 IC50 = 68 nM T28484 CJG9W1 86342431 IC50 = 3600 nM T28484 C9ZJ3Q 86342432 IC50 = 430 nM T28484 CC23YM 86342433 IC50 = 920 nM T28484 C3NIL0 86342434 IC50 = 50 nM T28484 CYZR27 86342435 IC50 = 51 nM T28484 C1W2BQ 90643994 IC50 = 85 nM T28484 CO03VM 90643995 IC50 > 6300 nM T28484 CE9ZK4 90643996 IC50 > 6300 nM T28484 CJWF68 90643997 IC50 = 390 nM T28484 CSFQ95 90643998 IC50 > 6300 nM T28484 CE3M0Q 90643999 IC50 > 6300 nM T28484 C5SBF7 90644000 IC50 > 6300 nM T28484 CI42NO 90644001 IC50 > 6300 nM T28484 C8QDX2 90644002 IC50 > 6300 nM T28484 CU6VR0 90644003 IC50 = 160 nM T28484 C9BUJ7 90644004 IC50 > 6300 nM T28484 C2S4RL 90644005 IC50 > 6300 nM T28484 C7Q6DK 90644006 IC50 > 6300 nM T28484 CQF0A2 90644007 IC50 > 6300 nM T28484 C8YC9V 90644008 IC50 > 6300 nM T28484 C8SXG7 90644009 IC50 > 6300 nM T28484 CB70HL 90644010 IC50 > 6300 nM T28484 CJC67A 90644011 IC50 > 6300 nM T28484 CAQF46 90644012 IC50 > 6300 nM T28484 C75EMH 90644013 IC50 = 4600 nM T28484 C28MTR 90644014 IC50 > 6300 nM T28484 CUN3W4 90644015 IC50 > 6300 nM T28484 C3JW6B 90644016 IC50 > 6300 nM T28484 CGM90T 118709485 IC50 = 44 nM T28484 CT6R9O 118721856 IC50 = 520 nM T28484 CWUL90 122195342 IC50 = 1060 nM T28484 CXSO48 122195343 IC50 = 306 nM T28484 C2BWQ7 122195344 IC50 = 238 nM T28484 CI24TL 122195345 IC50 = 160 nM T28484 CSN3F9 122195346 IC50 = 36 nM T28484 CI7MK5 122195347 IC50 = 8.6 nM T28484 CW81CB 122195348 IC50 = 12 nM T28484 CN69PC 122195349 IC50 = 1400 nM T28484 C3N2JL 122195350 IC50 > 20000 nM T28484 CSB5A6 122195351 IC50 > 20000 nM T28484 CYRN15 122195352 IC50 > 20000 nM T28484 CASH54 127035330 IC50 = 1460 nM T28484 C7I6KC 127037279 IC50 = 840 nM T28484 C9Z2CL 134133387 IC50 = 6800 nM T28484 C9GR4X 134141351 IC50 > 20000 nM T28484 C8HX3F 135981700 IC50 = 9000 nM T28484 C6KW0R 145954973 IC50 = 11390 nM T28484 C6HT9G 145962931 IC50 = 9030 nM T28484 C1ST4D 145978176 IC50 = 4860 nM T28484 CWAK78 145979859 IC50 = 41100 nM T28484 C15VPI 145982524 IC50 = 120000 nM T28484 C1QTO7 145982560 IC50 = 60000 nM T28484 CJ3CB4 145983009 IC50 = 20200 nM T28484 CA26IM 145983110 IC50 = 70000 nM T28484 C2AS3H 145983171 IC50 = 120000 nM T28484 CNHW71 145983379 IC50 = 71900 nM T28484 CV6O9Y 145983398 IC50 = 47800 nM T28484 C3XWO4 145983532 IC50 = 51000 nM T28484 CGYI36 145983831 IC50 = 133500 nM T28484 C5D7ZK 145984469 IC50 = 106200 nM T28484 C0V1ZO 145984507 IC50 = 42700 nM T28484 CJ5Z0S 145984542 IC50 = 13200 nM T28484 CP17GR 145984551 IC50 = 90000 nM T28484 CS62PR 145984570 IC50 = 39200 nM T28484 CGA0M2 145984674 IC50 = 17200 nM T28484 CVO4X7 145984986 IC50 = 27500 nM T28484 CL0X1V 145985314 IC50 = 62100 nM T28484 C2QZN6 145985512 IC50 = 128700 nM T28484 CH5V4P 145985905 IC50 = 90000 nM T28484 CWL1Z4 145985964 IC50 = 75000 nM T28484 C3QL0R 145985999 IC50 = 63300 nM T28484 CCTS70 145987224 IC50 = 59900 nM T28484 CTN4Q2 145990080 IC50 = 2200 nM T28484 CKSM25 145991640 IC50 = 53900 nM T28484 C3WQ7O 145992319 IC50 = 7500 nM T28484 CM5N9C 145993225 IC50 = 46900 nM T28484 D00HFV 11652296 IC50 = 11 nM T28484 D00OZN 23626453 IC50 = 7200 nM T28484 D00PRE 23625979 IC50 = 345 nM T28484 D00WOE 11254540 IC50 = 2002 nM T28484 D01ESV 23626139 IC50 = 716 nM T28484 D02HMN 46855212 IC50 = 870 nM T28484 D02LDY 11737887 IC50 = 7682 nM T28484 D02SGH 46244082 IC50 = 390 nM T28484 D05MQU 11695867 IC50 = 58 nM T28484 D05OMR 11299083 IC50 = 11000 nM T28484 D06HLH 46855216 IC50 = 1400 nM T28484 D08FXD 20228010 IC50 = 1500 nM T28484 D08RMK 11593788 IC50 = 1382 nM T28484 D09DGA 9196 IC50 = 4600 nM T28484 D09FZW 46855213 IC50 = 510 nM T28484 D09MSF 12462654 IC50 = 300 nM T28484 D09MXK 42611896 IC50 = 950 nM T28484 D09PLT 12117342 IC50 = 240 nM T28484 D0A9IB 23625978 IC50 = 3726 nM T28484 D0AV3M 11630239 IC50 = 57 nM T28484 D0CU4Q 24417 IC50 > 63000 nM T28484 D0D3FV 18504802 IC50 = 14000 nM T28484 D0E2KC 15541181 IC50 = 64 nM T28484 D0EC0B 44191658 IC50 = 7500 nM T28484 D0G1DW 11232325 Ki = 6.2 nM T28484 D0H3OP 138537 IC50 = 2800 nM T28484 D0H7ZS 23626454 IC50 = 10904 nM T28484 D0J9UC 11623295 IC50 = 140 nM T28484 D0JN0N 11695302 IC50 = 240 nM T28484 D0K7HV 11659042 IC50 = 54 nM T28484 D0M3VA 16034829 Ki < 1 nM T28484 D0M3ZV 504067 IC50 = 17000 nM T28484 D0M7KF 44191653 IC50 = 1600 nM T28484 D0MW5Z 24741169 IC50 = 11000 nM T28484 D0N5OD 9877863 IC50 = 5320 nM T28484 D0N8FU 46855214 IC50 = 3200 nM T28484 D0NJ8L 11595053 IC50 = 262 nM T28484 D0O5SA 10010225 IC50 = 3500 nM T28484 D0OF6C 12169809 IC50 = 210 nM T28484 D0OS3L 42611736 IC50 = 3300 nM T28484 D0P9ZN 46855064 IC50 = 8800 nM T28484 D0RO7K 19290 IC50 = 22000 nM T28484 D0S0JL 193613 IC50 > 63000 nM T28484 D0S7AY 276707 IC50 = 145000 nM T28484 D0T6MF 46855215 IC50 = 11000 nM T28484 D0TN1F 2782709 IC50 = 1649 nM T28484 D0TR0R 12169810 IC50 = 13000 nM T28484 D0V6CM 11593764 IC50 = 1600 nM T28484 D0W4GY 15541180 IC50 = 700 nM T28484 D0Y6IQ 49799223 IC50 = 5600 nM T28484 D0Z3KV 430297 IC50 = 22000 nM T73863 D0T5WK 4506 IC50 > 200000 nM T73863 D00SUC 74766595 IC50 = 35 nM T73863 D01WHH 90216982 IC50 = 1000 nM T73863 D03TKM 76901247 IC50 = 1100 nM T73863 D04KUD 56589666 IC50 < 500 nM T73863 D05CCY 77106319 IC50 < 100 nM T73863 D09NCT 53392492 IC50 = 4300 nM T73863 D0BK5N 56589667 IC50 < 500 nM T73863 D0G8QR 76282772 IC50 = 100 nM T73863 D0GH8J 90204862 IC50 = 54 nM T73863 D0HT9Q 77106317 IC50 = 199.53 nM T73863 D0K4LW 90205053 IC50 = 1000 nM T73863 CIC2K0 1048 Ki > 200000 nM T73863 CTXS46 70914 IC50 = 2070000 nM T73863 C0PU3Z 76559 Ki > 200000 nM T73863 CE73ZQ 78046 Ki > 200000 nM T73863 CT7CW5 144086 Ki > 200000 nM T73863 CF1MG5 338352 Ki > 200000 nM T73863 C1P0WX 344114 IC50 = 2810000 nM T73863 C76AMR 439391 IC50 = 79000 nM T73863 CT0H6S 439939 IC50 = 97000 nM T73863 C5K3ZJ 459531 IC50 = 630.96 nM T73863 C8B1QV 542717 Ki > 200000 nM T73863 CKJ28Z 555194 Ki > 200000 nM T73863 CX34DR 562549 Ki > 200000 nM T73863 C7MOV3 576286 Ki > 200000 nM T73863 CV4ZC0 584578 IC50 > 100000 nM T73863 CS4P5Z 688417 IC50 = 18600 nM T73863 C8M5EK 688418 IC50 = 54700 nM T73863 CMKP07 736587 IC50 < 1000 nM T73863 CHV9I2 762277 Ki > 200000 nM T73863 CZ8IW1 817743 IC50 > 100000 nM T73863 C89WXM 1273303 Ki > 200000 nM T73863 CP53HR 1398473 Ki > 200000 nM T73863 CEQ4V8 2723716 IC50 > 100000 nM T73863 CTSO67 2755894 Ki > 200000 nM T73863 CY3V0G 2784459 IC50 = 30000 nM T73863 CTH86O 2801750 Ki > 200000 nM T73863 CBMG93 4763332 IC50 = 165000 nM T73863 CIUB05 5513694 IC50 = 176000 nM T73863 CTC90M 6519698 IC50 = 1000 nM T73863 CCYF63 9942424 IC50 = 199.53 nM T73863 CF95UP 10909714 IC50 > 100000 nM T73863 CU1Y9B 11251979 Ki > 200000 nM T73863 CD6JS2 13047427 Ki > 200000 nM T73863 C84NIM 13413393 IC50 = 100000 nM T73863 C8NG1A 13973357 Ki > 200000 nM T73863 C1PSK2 13973362 Ki > 200000 nM T73863 C0N6VT 14536434 Ki > 200000 nM T73863 CR52CA 14638329 Ki > 200000 nM T73863 C6RG4X 15179913 Ki > 200000 nM T73863 CTVD27 16773856 IC50 = 98000 nM T73863 C5R0VE 16790848 IC50 = 126000 nM T73863 CA2K7C 19623349 IC50 = 387000 nM T73863 CB1ZF9 19624675 IC50 = 58000 nM T73863 CMT92U 21766412 Ki > 200000 nM T73863 C8VQ2R 22042185 Ki > 200000 nM T73863 CCAM68 22959876 IC50 = 34000 nM T73863 CKQ14T 23610474 Ki > 200000 nM T73863 CF47JU 25138011 IC50 = 3500 nM T73863 C5O1XD 26967300 IC50 = 676000 nM T73863 C7X3WA 28330466 IC50 > 100000 nM T73863 C7OJ5E 46899602 IC50 = 2700 nM T73863 CUMF70 46899605 IC50 = 1500 nM T73863 C2DBN5 46899607 IC50 = 1000 nM T73863 C3G4QK 46899609 IC50 = 1600 nM T73863 C24GUR 46899759 IC50 = 5200 nM T73863 C6ZR3Y 46899761 IC50 = 8800 nM T73863 CLK96Z 46899763 IC50 = 2000 nM T73863 CBOM64 46899765 IC50 = 15000 nM T73863 C9ENX8 46899767 IC50 = 1300 nM T73863 CF2QL4 46899769 IC50 = 1700 nM T73863 CW10BJ 46901089 IC50 = 10000 nM T73863 C6Z1NU 46901246 IC50 = 74000 nM T73863 CUN94R 50999408 IC50 = 507000 nM T73863 CM07QJ 53380011 IC50 = 51000 nM T73863 C2HXA1 53380104 IC50 = 61000 nM T73863 C8CMI9 56766349 IC50 = 2320000 nM T73863 C6QTC3 64393791 IC50 = 316.23 nM T73863 CM9Y5X 64394359 IC50 = 1258.93 nM T73863 CELF46 64394751 IC50 = 398.11 nM T73863 C8K7LG 64395323 IC50 = 316.23 nM T73863 CVYI52 70682586 Ki > 200000 nM T73863 C0HM6A 70682588 Ki > 200000 nM T73863 C6BXR0 70684674 Ki > 200000 nM T73863 CZM97K 70684675 Ki > 200000 nM T73863 C6KM4Y 70684676 Ki > 200000 nM T73863 C81APE 70686821 Ki > 200000 nM T73863 C7SI8G 70688900 Ki > 200000 nM T73863 CAYC62 70688901 Ki > 200000 nM T73863 C5BA6D 70688902 Ki > 200000 nM T73863 C9HTX1 70690990 Ki > 200000 nM T73863 C0DO2G 70690991 Ki > 200000 nM T73863 CDQ5H7 70693123 Ki > 200000 nM T73863 CI1M5B 70695173 Ki > 200000 nM T73863 CB3VJ9 70695181 Ki > 200000 nM T73863 CB80OC 70695182 Ki > 200000 nM T73863 CM4J9D 70695183 Ki > 200000 nM T73863 CJK98Q 70695184 Ki > 200000 nM T73863 CB46OW 70697226 Ki > 200000 nM T73863 CI19FA 70697227 Ki > 200000 nM T73863 C14GIV 71735687 IC50 = 81000 nM T73863 CM02VN 71735839 IC50 = 32000 nM T73863 C4WS1H 71735840 IC50 = 22000 nM T73863 CT4YO5 71735841 IC50 = 78000 nM T73863 C2ZFM8 71735842 IC50 > 120000 nM T73863 CI5W0K 71735843 IC50 = 83000 nM T73863 C6GDP2 71765680 IC50 = 199.53 nM T73863 CN53LH 71765996 IC50 = 6309.57 nM T73863 C2RT5O 71765999 IC50 = 63095.73 nM T73863 C6DXR4 71766146 IC50 = 6309.57 nM T73863 CDT16O 71766431 IC50 = 125.89 nM T73863 CO5TU3 71766576 IC50 = 1995.26 nM T73863 COCF38 71767872 IC50 = 31622.78 nM T73863 CYF8O7 71767874 IC50 = 40000 nM T73863 CFY18G 73333510 IC50 = 110000 nM T73863 CN5B4O 73352277 IC50 = 55000 nM T73863 C68RKH 76310231 IC50 = 1200 nM T73863 CO1EN3 76317452 IC50 = 70 nM T73863 CT5FZ8 76321184 IC50 = 4500 nM T73863 C6XRT0 76321186 IC50 = 2700 nM T73863 CKB5O9 76328366 IC50 = 2500 nM T73863 CUNK03 76335652 IC50 = 3100 nM T73863 C4HXD2 76901248 IC50 = 1100 nM T73863 C4VGX7 76901615 IC50 = 380 nM T73863 CZC7E1 76901616 IC50 = 660 nM T73863 CC5WE1 76901618 IC50 = 2700 nM T73863 CA79XV 76901619 IC50 = 1800 nM T73863 CM2L1V 76901620 IC50 = 410 nM T73863 CLM1B2 77107119 IC50 = 12 nM T73863 CYOA89 77107120 IC50 > 2000 nM T73863 C16PNL 77107121 IC50 = 8 nM T73863 C6IJN1 78426128 IC50 = 1000 nM T73863 CX23ZP 78426670 IC50 > 2500 nM T73863 CMR52S 78426698 IC50 = 2000 nM T73863 CKXW73 78427224 IC50 > 2500 nM T73863 CFPV20 78972837 IC50 = 1210000 nM T73863 C9IMX6 81750118 IC50 = 316.23 nM T73863 C63ATV 81750201 IC50 = 79.43 nM T73863 CHY73I 81750365 IC50 = 158.49 nM T73863 CE6OT2 81750629 IC50 = 31622.78 nM T73863 C21MQV 81750712 IC50 = 630.96 nM T73863 CQG60A 81750714 IC50 <= 100 nM T73863 CM9P8V 81750970 IC50 = 199.53 nM T73863 C69YUM 81751142 IC50 = 125.89 nM T73863 CW47ZA 83454396 IC50 = 5200 nM T73863 C17WNZ 83698744 IC50 = 501.19 nM T73863 CYG63D 86222684 Ki > 200000 nM T73863 CS4Q1F 86268882 IC50 < 100 nM T73863 CRQ51Z 86346639 IC50 < 100 nM T73863 CZ9DC6 86725498 IC50 = 6200 nM T73863 C8WA4M 86725535 IC50 = 5 nM T73863 C8MGN0 86725568 IC50 = 14 nM T73863 CW9F0K 89564218 IC50 < 1000 nM T73863 CCI08H 89825587 IC50 <= 100 nM T73863 C83TUW 89825693 IC50 <= 100 nM T73863 CT46KN 90094283 IC50 = 100 nM T73863 CG4BZ9 90094442 IC50 < 100 nM T73863 C9IYE0 90204662 IC50 = 38 nM T73863 CHV05N 90204861 IC50 = 68 nM T73863 C6PI4M 90204893 IC50 = 2900 nM T73863 CIY20E 90204966 IC50 = 280 nM T73863 CK6L5M 90205111 IC50 = 560 nM T73863 C5ST7H 90205231 IC50 = 1100 nM T73863 CQV07L 90205291 IC50 = 3600 nM T73863 CJ5E4U 90205326 IC50 = 78 nM T73863 C5W7FL 90205353 IC50 = 19 nM T73863 CR21SC 90205356 IC50 = 2900 nM T73863 CM2NA1 90205425 IC50 = 24 nM T73863 CB7Z0A 90205426 IC50 = 74 nM T73863 CN9I0J 90205512 IC50 = 490 nM T73863 C2T4RD 90205719 IC50 = 260 nM T73863 C9H8PV 90211058 IC50 = 310 nM T73863 C1GBT5 90225370 IC50 = 100 nM T73863 CFP3G4 90253472 IC50 = 100 nM T73863 CPUK85 90253505 IC50 = 6 nM T73863 CFX8E0 90407594 IC50 > 10000 nM T73863 CJ9OZ4 90407809 IC50 = 1000 nM T73863 C5LDR2 90407841 IC50 = 100 nM T73863 C2NA5I 91801131 IC50 = 6309.57 nM T73863 CQY0K3 91938043 IC50 < 250 nM T73863 C10RDJ 101882871 IC50 = 15848.93 nM T73863 C86LNW 101882872 IC50 > 100000 nM T73863 C2S1AO 110264830 IC50 = 13300 nM T73863 C4FPD3 112726150 IC50 > 100000 nM T73863 C5OUS0 114286469 IC50 <= 100 nM T73863 C12QPH 114288702 IC50 = 31622.78 nM T73863 CT04PB 118420691 IC50 < 250 nM T73863 CPSD31 118420829 IC50 < 250 nM T73863 CU94QR 118421047 IC50 > 2500 nM T73863 CH6FX3 118421371 IC50 < 250 nM T73863 C6YT2Q 118598059 EC50 = 1.3 nM T73863 C7TBE9 118908379 IC50 = 1900 nM T73863 CJVK69 119081409 IC50 = 4100 nM T73863 C5IZD1 122181577 IC50 = 55000 nM T73863 CY3CG7 122181578 IC50 > 100000 nM T73863 CSR0K5 122181579 IC50 = 63000 nM T73863 CQ57MD 122181580 IC50 = 6500 nM T73863 CQ83MR 122181581 IC50 = 62000 nM T73863 C4GU9P 122181582 IC50 = 76000 nM T73863 CRM93S 122181583 IC50 = 37000 nM T73863 CU57QX 122181584 IC50 = 43000 nM T73863 CIM8C2 122181585 IC50 = 65000 nM T73863 CQA0H7 122181586 IC50 > 100000 nM T73863 C9QVZ5 122181587 IC50 > 100000 nM T73863 CJQ91K 122181588 IC50 = 83000 nM T73863 C8E2KI 122191450 IC50 = 3162.28 nM T73863 C75JVN 122191451 IC50 = 10000 nM T73863 C3YX7W 122191453 IC50 = 6309.57 nM T73863 C3IBR8 122191455 IC50 = 5011.87 nM T73863 C59KNQ 122191457 IC50 = 39810.72 nM T73863 CM5X8J 122191459 IC50 = 39810.72 nM T73863 C7ASR0 122191460 IC50 > 100000 nM T73863 CRI6J4 122191461 IC50 > 100000 nM T73863 CAS4H6 122191462 IC50 = 15848.93 nM T73863 C9J6LX 122191463 IC50 = 15848.93 nM T73863 C75NJO 122191464 IC50 = 10000 nM T73863 C50VYK 122191465 IC50 = 31622.78 nM T73863 CSKY20 122191466 IC50 = 79432.82 nM T73863 CS3L8H 122191467 IC50 = 1584.89 nM T73863 CZ2NV1 122191468 IC50 = 12589.25 nM T73863 CYTW93 122191469 IC50 = 7943.28 nM T73863 CZV45H 122191470 IC50 = 19952.62 nM T73863 CF6I2N 122191471 IC50 = 39810.72 nM T73863 CZU02B 122191472 IC50 = 7943.28 nM T73863 CE27AS 122191473 IC50 = 19952.62 nM T73863 CAJ28B 122191475 IC50 = 31622.78 nM T73863 C36PDK 122191476 IC50 = 39810.72 nM T73863 CQ04FW 122191477 IC50 = 15848.93 nM T73863 C12OHA 122191478 IC50 = 15848.93 nM T73863 CL2K0J 122191479 IC50 = 19952.62 nM T73863 CT6HG3 122191480 IC50 = 19952.62 nM T73863 CK7LD6 122191481 IC50 = 19952.62 nM T73863 CMJ72N 122191482 IC50 = 25118.86 nM T73863 C6H2YQ 122383780 IC50 = 5000 nM T73863 CT2UZ4 125377518 IC50 = 3900 nM T73863 CV6H7C 127028789 IC50 >= 100000 nM T73863 CB8GP9 127029091 IC50 = 25118.86 nM T73863 CIJ0G6 127030272 IC50 < 250 nM T73863 C6KT5A 127030498 IC50 = 310000 nM T73863 C63NWD 127030711 IC50 < 1000 nM T73863 CXF0U5 127030712 IC50 < 1000 nM T73863 CZ2M7U 127030808 IC50 = 125.89 nM T73863 CN16WB 127030937 IC50 < 100 nM T73863 CO4UE5 127031137 IC50 = 15000 nM T73863 CBC7G1 127032036 IC50 = 1258.93 nM T73863 CHO3V7 127032343 IC50 = 1584.89 nM T73863 CB6LF9 127032423 IC50 = 600 nM T73863 C8U9DH 127032712 IC50 = 8500 nM T73863 CDC17F 127032730 IC50 < 100 nM T73863 C5SKT0 127032945 IC50 = 15848.93 nM T73863 CW14UR 127032962 IC50 = 630.96 nM T73863 CL38FP 127033048 IC50 < 100 nM T73863 C2EY1K 127033166 IC50 < 250 nM T73863 CID1E9 127034046 IC50 < 250 nM T73863 C4L1PZ 135567036 IC50 = 6000 nM T73863 CT4O5U 135567037 Ki = 682.9 nM T73863 CC4H1N 135567038 IC50 = 5000 nM T73863 C3LG4V 135567039 IC50 = 8300 nM T73863 CQBH95 135567040 IC50 = 1200 nM T73863 CP6IH9 135567041 Ki = 43.2 nM T73863 C8HMG2 135567042 IC50 = 140 nM T73863 CIW61V 135567106 IC50 = 1995.26 nM T73863 CH2D8B 135567124 IC50 = 398.11 nM T73863 CO1F4A 135567128 IC50 = 501.19 nM T73863 CT0DW5 136048747 IC50 < 100 nM T73863 CXW0S7 136048748 IC50 < 100 nM T73863 CJ91RY 136048749 IC50 < 100 nM T73863 CI4X6R 136053672 IC50 = 1995.26 nM T73863 CO6A0C 136053673 IC50 = 2511.89 nM T73863 CD9F1K 136053674 IC50 = 630.96 nM T73863 CE9R0F 136053675 IC50 = 630.96 nM T73863 CIZV97 136053676 IC50 = 398.11 nM T73863 CE1SW8 136053677 IC50 = 630.96 nM T73863 C8S7CR 136053678 IC50 = 501.19 nM T73863 C3V1SD 136053679 IC50 = 398.11 nM T73863 CMW30T 136053680 IC50 = 630.96 nM T73863 C97FZE 136053681 IC50 = 501.19 nM T73863 CQND25 136053682 IC50 = 7943.28 nM T73863 C6IJ5M 136053683 IC50 = 2000 nM T73863 CNY5T7 136053684 IC50 = 398.11 nM T73863 CV57DW 136053685 IC50 = 199.53 nM T73863 CBGO86 136053686 IC50 = 501.19 nM T73863 C3K1OC 136053687 IC50 = 501.19 nM T73863 CZ80GB 136053688 IC50 = 3162.28 nM T73863 CN56RV 136053689 IC50 = 3162.28 nM T73863 C8HOP7 136053690 IC50 = 1995.26 nM T73863 CN4L7Q 136053691 IC50 = 630.96 nM T73863 CO17WM 136053692 IC50 = 1000 nM T73863 C6OJ3M 136053693 IC50 = 794.33 nM T73863 C5ANQ0 136053694 IC50 = 3162.28 nM T73863 CG13YI 136053695 IC50 = 12589.25 nM T73863 C4EW6T 136053696 IC50 = 1995.26 nM T73863 C5Q9HO 136053697 IC50 = 7943.28 nM T73863 CL3DH6 136053700 IC50 = 4600 nM T73863 C8BAQ6 136053701 IC50 = 460 nM T73863 C3I0DN 136053702 IC50 = 430 nM T73863 CHYC17 136053703 IC50 = 170 nM T73863 CW5FY8 136053704 IC50 = 69 nM T73863 C0DB1S 136053705 IC50 = 1020 nM T73863 C63EQY 136053706 IC50 = 770 nM T73863 C7ALO8 136053707 IC50 = 560 nM T73863 C86NDI 136053708 IC50 = 2500 nM T73863 CR6QH4 136164086 IC50 = 19952.62 nM T73863 CM2VE8 136165229 IC50 = 1900 nM T73863 CU10SL 136258480 IC50 = 450 nM T73863 C2V6MX 136644692 IC50 > 100000 nM T73863 C1H9NK 136959977 IC50 = 100 nM T73863 C1ANF3 138518187 IC50 > 25000 nM T73863 C6LWR4 145963760 IC50 = 151 nM T73863 C0RPS4 145964567 IC50 = 55 nM T73863 C3U8OD 145966600 IC50 = 466 nM T73863 CM9X8H 145967298 IC50 = 12 nM T73863 C9U5TQ 145967792 IC50 = 23 nM T73863 CB97SG 145968018 IC50 = 53 nM T73863 CT5MO6 145971004 IC50 = 154 nM T73863 CK9V5O 145972063 IC50 = 27 nM T73863 CS5FM7 145974200 EC50 = 19 nM T73863 CC8KI6 145976146 IC50 = 23 nM T73863 C1AUN0 145976182 IC50 = 17 nM T73863 CKU0D3 145976400 IC50 = 173 nM T73863 CQ4E0O 145977225 IC50 = 65 nM T73863 CIQ6Y7 145977327 IC50 = 2.2 nM T73863 C5TBS2 145977546 IC50 = 46 nM T73863 CL2FR4 145978064 IC50 = 22 nM T73863 C8OL2Q 145978411 IC50 = 164 nM T73863 CA8UD0 145978535 IC50 = 38 nM T73863 D07IOY 10365 Ki = 2.2 nM T73863 D08IZY 3080614 IC50 = 430000 nM T73863 D0B2WZ 15331 IC50 = 2500000 nM T73863 D0M7DC 574310 Ki > 200000 nM T73863 D0X5US 459617 IC50 = 600 nM T65483 CMU34O 9813856 IC50 > 50000 nM T65483 CF5A3T 9837547 IC50 > 50000 nM T65483 CQ6HP2 9857137 IC50 > 50000 nM T65483 CHI95J 9926432 IC50 > 50000 nM T65483 C9WT3L 9942902 IC50 > 50000 nM T65483 CM1A0D 9943447 IC50 > 50000 nM T65483 CW28EQ 9966944 IC50 > 50000 nM T65483 C6FQ0R 10465893 IC50 > 50000 nM T65483 D06LNX 3858 IC50 > 50000 nM T33754 D03VPC 2754 IC50 = 190 nM T33754 D05MQK 110635 IC50 > 10000 nM T33754 D0C4HG 3033825 IC50 = 8 nM T33754 D0C9SY 135400189 IC50 = 2100 nM T33754 D0D1HW 135409400 IC50 = 50 nM T33754 D0E0SW 53708 IC50 = 14000 nM T33754 D0F8RA 2153 IC50 = 240000 nM T33754 D0F9GE 3108 IC50 = 43000 nM T33754 D0L0ZF 5663 IC50 = 6200 nM T33754 D0Y9ZE 4197 Ki = 150 nM T33754 D0Z7ZM 135398744 IC50 = 7000 nM T33754 D01LCC 17754438 IC50 = 1300 nM T33754 D08HKT 5362399 IC50 = 300 nM T33754 D0LI1C 44469321 IC50 > 10000 nM T33754 D0O1IM 58298318 IC50 = 630 nM T33754 D0SM0W 44591583 IC50 = 6400 nM T33754 D0T5PO 5092 IC50 > 10000 nM T33754 D0X0PP 59351313 IC50 > 30000 nM T33754 D07EUB 46200734 IC50 = 1820 nM T33754 D00DBE 9865514 IC50 = 35800 nM T33754 D00SPK 23665864 IC50 > 100000 nM T33754 D00YPW 135399235 IC50 = 133000 nM T33754 D01QUF 9842576 Ki > 100000 nM T33754 D02EMR 151170 IC50 > 3162.28 nM T33754 D05VLN 55690 IC50 = 31622.78 nM T33754 D07FHZ 5087 IC50 > 300000 nM T33754 D08FOX 55263 IC50 = 8600 nM T33754 D08NXX 5487281 IC50 = 10 nM T33754 D09SFV 3973 IC50 = 100000 nM T33754 D09UMA 55918 IC50 = 3400 nM T33754 D0BK6B 3021729 IC50 = 260 nM T33754 D0F0CS 5723 IC50 = 110 nM T33754 D0Y6HV 187079 IC50 = 50 nM T33754 CVQ0G5 1348 Ki = 16000 nM T33754 CO2Y3R 3698 IC50 = 16000 nM T33754 CX43RE 4823 IC50 = 19000 nM T33754 CH8J2B 4977 Ki = 1000000 nM T33754 CCJ8F0 5353 IC50 = 500000 nM T33754 C3B8VG 5369 IC50 > 10000 nM T33754 CJ02EG 41946 Ki = 1400 nM T33754 CA5Q8Y 58575 IC50 = 17000 nM T33754 CJ5R9Z 60867 IC50 = 1500 nM T33754 C1OJE8 65934 IC50 = 1600 nM T33754 CZ39NL 127770 IC50 = 37000 nM T33754 CGA17S 127779 Ki = 35000 nM T33754 C54IRL 129517 IC50 = 1500 nM T33754 CB9XD5 129826 IC50 = 100 nM T33754 C3B1GP 130152 IC50 = 47 nM T33754 C3FRX9 131989 IC50 = 380000 nM T33754 COK69D 156890 IC50 = 390000 nM T33754 CH2P8A 158961 Ki = 1200000 nM T33754 CVN23X 158962 Ki = 1100000 nM T33754 CGO1D9 184661 IC50 = 125.89 nM T33754 C4IEB6 205981 Ki = 217000 nM T33754 C8FWD2 317789 IC50 = 2511.89 nM T33754 C8EFH4 349956 IC50 = 101000 nM T33754 CG7Q1D 589674 IC50 = 18800 nM T33754 C6FCR1 3015712 IC50 = 138000 nM T33754 C1UNV3 4197712 IC50 = 14000 nM T33754 CBS67I 5271722 IC50 = 61000 nM T33754 CR5GH1 5284402 IC50 = 80 nM T33754 CE5VJ9 5362132 IC50 = 550 nM T33754 CO8NK7 5487388 IC50 = 18 nM T33754 CYO52K 5487415 IC50 = 0.4 nM T33754 COPL36 5492199 IC50 = 24 nM T33754 CSQ14B 5492217 IC50 = 20 nM T33754 C7BQ1N 5492386 IC50 = 1 nM T33754 CXDJ97 5746185 IC50 = 300 nM T33754 C8ZFX6 6624932 IC50 = 160000 nM T33754 CAYS61 6918354 IC50 = 290 nM T33754 CB40PM 6918356 IC50 = 1800 nM T33754 CR0NJ7 6918510 IC50 = 27000 nM T33754 CFJ62Y 9799389 IC50 > 10000 nM T33754 C3EOU7 9799418 IC50 > 3162.28 nM T33754 C87ERL 9806003 IC50 = 251.19 nM T33754 CHK3Z5 9806981 IC50 = 199.53 nM T33754 C0F5WH 9816616 IC50 = 2000 nM T33754 CXF0J7 9818343 IC50 = 12000 nM T33754 C1CXA5 9818702 IC50 = 380000 nM T33754 CSOX21 9819114 IC50 > 3000 nM T33754 C1MN3A 9821924 IC50 = 2220 nM T33754 C0K3SA 9825739 IC50 > 100000 nM T33754 C7B1PO 9826435 IC50 = 51600 nM T33754 CKG34S 9828282 IC50 = 501.19 nM T33754 CKOT49 9829555 IC50 = 100 nM T33754 C3ZNU4 9850384 IC50 = 79.43 nM T33754 CFV1Q4 9852021 IC50 > 3162.28 nM T33754 C8QJ4D 9859958 IC50 > 100000 nM T33754 C3HJB5 9867688 IC50 > 3162.28 nM T33754 CDW03H 9867844 IC50 > 3162.28 nM T33754 CVP6S0 9869611 IC50 = 79.43 nM T33754 CF18MC 9874535 IC50 > 100000 nM T33754 C7XYK6 9881656 IC50 > 100000 nM T33754 CQJ71T 9887909 IC50 > 3162.28 nM T33754 CY65BZ 9894329 IC50 = 199.53 nM T33754 CD6IG8 9894586 IC50 > 100000 nM T33754 CET1I4 9906369 IC50 > 20000 nM T33754 CMBO89 9912467 IC50 = 330 nM T33754 C81LSK 9928390 IC50 > 100000 nM T33754 CRT85B 9953239 IC50 = 80 nM T33754 COS23J 9956462 IC50 = 199.53 nM T33754 C19FKZ 9958988 IC50 > 3162.28 nM T33754 C4P8WX 9959207 IC50 = 31.62 nM T33754 CQ40MX 9981320 IC50 = 2400 nM T33754 C39LZS 9999105 IC50 = 30 nM T33754 CFPR64 9999276 IC50 > 10000 nM T33754 CKP7I8 10014043 IC50 = 350 nM T33754 C34ZPX 10014479 IC50 = 560 nM T33754 CXQ0V1 10016898 IC50 = 2000 nM T33754 C4ST7G 10017729 IC50 = 400 nM T33754 C3R8DT 10036672 IC50 = 4200 nM T33754 CHL52O 10037253 IC50 = 230 nM T33754 CMAT67 10038096 IC50 = 78 nM T33754 CJ1Q7Z 10040540 IC50 = 15000 nM T33754 CGXS34 10043016 IC50 = 5900 nM T33754 CH0YG4 10043540 IC50 = 37 nM T33754 CGX7W1 10064431 IC50 = 18000 nM T33754 C12KAB 10065195 IC50 = 850 nM T33754 C2L8MI 10068486 IC50 > 3162.28 nM T33754 CJA37O 10082617 IC50 = 22 nM T33754 CQMC42 10083083 IC50 = 180 nM T33754 C2N4IZ 10084561 IC50 = 12.59 nM T33754 C6QVN7 10104952 IC50 = 1400 nM T33754 COB5N2 10105100 IC50 = 2800 nM T33754 C8SNV1 10105196 IC50 = 160 nM T33754 CT0A4J 10113055 IC50 = 299 nM T33754 CPWL59 10113972 IC50 = 1060 nM T33754 C2MGJ7 10117650 IC50 = 580 nM T33754 CG8RW2 10142576 IC50 = 2970 nM T33754 C89DXP 10181676 IC50 = 2710 nM T33754 C8V6FE 10225063 IC50 = 42 nM T33754 CAS6F9 10228849 IC50 = 23300 nM T33754 CZ1Y8D 10232923 IC50 > 100000 nM T33754 C1TZ0Y 10242216 IC50 = 5300 nM T33754 CNF1Z7 10243366 IC50 = 1600 nM T33754 C41REA 10243444 IC50 = 23 nM T33754 C1XL2R 10247726 IC50 = 24000 nM T33754 CK23EJ 10261617 IC50 = 960 nM T33754 C7GTC0 10264205 IC50 > 10000 nM T33754 CJQ89G 10266192 IC50 > 200000 nM T33754 CUE72P 10314633 IC50 = 2000 nM T33754 CB71WD 10322207 IC50 = 16 nM T33754 C86USM 10326035 IC50 > 3162.28 nM T33754 CF6YU1 10329832 IC50 = 3100 nM T33754 CP1M5H 10342086 IC50 > 100000 nM T33754 C1Z6TS 10352208 IC50 = 3700 nM T33754 CC14IS 10354139 IC50 = 230 nM T33754 CU45BF 10354140 IC50 = 69 nM T33754 CZ6X9Y 10391444 IC50 = 290 nM T33754 CMR4H3 10398747 IC50 = 100 nM T33754 CU32AZ 10411395 IC50 > 3162.28 nM T33754 C94CHO 10421765 IC50 = 1400 nM T33754 CY6B3J 10422444 IC50 = 28000 nM T33754 C43YLO 10422686 IC50 = 330 nM T33754 CEOK50 10428730 IC50 < 10000 nM T33754 C3WG2D 10432384 IC50 > 3162.28 nM T33754 C1OG0Y 10443570 IC50 = 2200 nM T33754 C60KSF 10444558 IC50 = 67 nM T33754 CF5O8D 10446136 IC50 = 1850 nM T33754 C23HSK 10451184 IC50 > 100000 nM T33754 CHQ38X 10455790 IC50 > 100000 nM T33754 CH2B6U 10455813 IC50 = 2400 nM T33754 C5WAM6 10465078 IC50 = 1420 nM T33754 CN40VQ 10465933 IC50 = 62 nM T33754 C0XW2I 10469627 IC50 > 3000000 nM T33754 C5CI3G 10479468 IC50 = 90 nM T33754 CZ92DR 10481735 IC50 = 6030 nM T33754 CA24TW 10491646 IC50 > 100000 nM T33754 C68VBD 10492653 IC50 > 100000 nM T33754 C3PKX6 10492654 IC50 > 100000 nM T33754 C5JPK7 10494678 IC50 > 200000 nM T33754 C2OP8L 10497499 IC50 = 8500 nM T33754 CTUW75 10503944 IC50 = 320 nM T33754 CMR6A4 10504383 IC50 = 80000 nM T33754 C6GS9R 10506218 IC50 > 100000 nM T33754 C4CN0V 10508072 IC50 > 100000 nM T33754 CW7T6I 10515565 IC50 > 100000 nM T33754 CPWU60 10524067 IC50 = 20000 nM T33754 CH4LZ1 10525677 IC50 = 86800 nM T33754 CR8SN9 10526455 IC50 > 100000 nM T33754 C9WSE6 10528313 IC50 = 2900 nM T33754 CZ6T2C 10536740 IC50 > 100000 nM T33754 CCG53Q 10541661 IC50 = 77000 nM T33754 CLI1R7 10543311 IC50 > 200000 nM T33754 C6M0ZQ 10545256 IC50 = 3500 nM T33754 CP63QK 10547069 IC50 = 18000 nM T33754 C7G1BH 10547592 IC50 > 100000 nM T33754 CP0JT2 10550927 IC50 > 100000 nM T33754 C7ID5Q 10552011 IC50 = 82000 nM T33754 CQW79N 10554042 IC50 = 50000 nM T33754 C4V8OI 10563356 IC50 > 100000 nM T33754 C5WMZ0 10563923 IC50 = 30000 nM T33754 CYUJ54 10564633 IC50 > 200000 nM T33754 C1R0HE 10567025 IC50 > 200000 nM T33754 CKUS20 10567758 IC50 > 200000 nM T33754 C7K1QW 10571952 IC50 > 100000 nM T33754 CY9P5W 10575733 IC50 = 60 nM T33754 C8V2KW 10576728 IC50 = 46000 nM T33754 C20EPT 10577926 IC50 = 4500 nM T33754 C7Z9YF 10579873 IC50 > 100000 nM T33754 C3Y8JH 10590134 IC50 = 97000 nM T33754 CW0LN4 10593644 IC50 > 200000 nM T33754 C57HYA 10600864 IC50 = 16000 nM T33754 CMNU92 10602385 IC50 = 10600 nM T33754 CS2Q1U 10602534 IC50 > 100000 nM T33754 CSPY93 10603533 IC50 > 100000 nM T33754 CJ7CU4 10603606 IC50 = 34 nM T33754 CUTK97 10610142 IC50 = 68000 nM T33754 C5LVM2 10613420 IC50 > 100000 nM T33754 CK3GR5 10624131 IC50 = 400 nM T33754 CZIQ04 10625498 IC50 = 77000 nM T33754 CN4T7O 10625920 IC50 > 100000 nM T33754 C21CUM 10626417 IC50 > 100000 nM T33754 C1O4KV 10626842 IC50 > 100000 nM T33754 C25WRZ 10627119 IC50 = 170 nM T33754 CCB7D3 10639948 IC50 = 6000 nM T33754 CF1UR8 10640268 IC50 = 5000 nM T33754 CB3R6M 10644497 IC50 = 90000 nM T33754 CUZN30 10646721 IC50 = 70000 nM T33754 CNK65G 10646809 IC50 = 2000 nM T33754 CKNA14 10648008 IC50 = 250 nM T33754 C0I4FA 10648358 IC50 = 10300 nM T33754 CP8UX9 10649414 IC50 = 58200 nM T33754 C3XAK7 10650055 IC50 > 100000 nM T33754 CE65JO 10650764 IC50 > 100000 nM T33754 CNP1D9 10651107 IC50 > 100000 nM T33754 CJ5XI4 10651803 IC50 > 100000 nM T33754 CP2B0V 10660654 IC50 = 42000 nM T33754 CY25HA 10661817 IC50 = 58000 nM T33754 CP1CJ3 10663161 IC50 > 200000 nM T33754 CR47SU 10665209 IC50 = 4.9 nM T33754 C09ROH 10668502 IC50 > 100000 nM T33754 CB9Y7A 10669693 IC50 = 2000 nM T33754 CFM5N1 10673963 IC50 > 100000 nM T33754 C9FR7P 10674875 IC50 > 100000 nM T33754 C2Y5HF 10675032 IC50 = 490 nM T33754 C6T4ZW 10687037 IC50 = 14000 nM T33754 C5KXY7 10688351 IC50 > 200000 nM T33754 CHB93E 10690761 IC50 = 200000 nM T33754 CV6WT3 10692240 IC50 > 100000 nM T33754 C6LR4V 10694878 IC50 > 100000 nM T33754 CV0H5I 10696630 IC50 = 54700 nM T33754 C1B3WP 10696971 IC50 = 3200 nM T33754 CI6ON5 10698519 IC50 = 100 nM T33754 C40GRD 10704663 IC50 = 331000 nM T33754 C23WGX 10706416 IC50 > 100000 nM T33754 C59SWD 10709216 IC50 = 43000 nM T33754 C8CM0J 10711062 IC50 = 44000 nM T33754 C8UHE3 10717022 IC50 = 9000 nM T33754 CDMP96 10717370 IC50 = 20000 nM T33754 CEW0L8 10718244 IC50 > 100000 nM T33754 CU53RA 10718426 IC50 = 18000 nM T33754 CCI8R7 10729204 IC50 > 100000 nM T33754 CF7L2E 10732847 IC50 = 29000 nM T33754 CS2ZA3 10734331 IC50 > 200000 nM T33754 C5IKL9 10734997 IC50 = 20000 nM T33754 C7JN8X 10739699 IC50 = 3500 nM T33754 CO39UQ 10744528 IC50 = 22200 nM T33754 C3X8UM 10754735 IC50 = 80000 nM T33754 CDPZ05 10758281 IC50 > 200000 nM T33754 C28FLE 10762239 IC50 = 18000 nM T33754 CINX82 10763354 IC50 = 80000 nM T33754 C3R8TI 10764856 IC50 = 28800 nM T33754 CFJL61 10768238 IC50 = 41 nM T33754 C51XRM 10776762 IC50 > 300000 nM T33754 C35YPM 10779997 IC50 > 200000 nM T33754 CO08EH 10780064 IC50 = 45000 nM T33754 CSN64H 10783300 IC50 > 200000 nM T33754 CEV60G 10783489 IC50 = 18000 nM T33754 COF0E3 10783717 IC50 > 1000 nM T33754 CKEV02 10786459 IC50 > 200000 nM T33754 CQMF39 10787820 IC50 > 100000 nM T33754 CLM42P 10788651 IC50 = 8000 nM T33754 C92SMD 10789583 IC50 = 53900 nM T33754 C19EHR 10791038 IC50 > 100000 nM T33754 CXWY95 10792119 IC50 > 100000 nM T33754 C6C5AD 10792156 IC50 > 100000 nM T33754 C2KUF1 10792829 IC50 > 100000 nM T33754 C1K4AN 10792853 IC50 > 100000 nM T33754 C9YFH4 10805458 IC50 > 200000 nM T33754 C24LPM 10810360 IC50 = 12000 nM T33754 CDL73U 10810934 IC50 > 100000 nM T33754 CAF1X8 10812634 IC50 > 100000 nM T33754 CW07PN 10814053 IC50 = 48600 nM T33754 CA9UW6 10816539 IC50 = 81 nM T33754 C4T8PS 10816641 IC50 > 100000 nM T33754 CX1B4U 10817302 IC50 = 60000 nM T33754 C49GKH 10826458 IC50 > 200000 nM T33754 CG5M7O 10827879 IC50 = 58000 nM T33754 CT8AK4 10830480 IC50 = 64000 nM T33754 COHP57 10833764 IC50 > 100000 nM T33754 CT2F6P 10835916 IC50 = 8000 nM T33754 C0QY8J 10837144 IC50 = 48500 nM T33754 CZMB59 10840332 IC50 > 100000 nM T33754 C5MTK7 10840471 IC50 > 100000 nM T33754 C2IWD7 10840815 IC50 > 100000 nM T33754 CR50XV 10841036 IC50 = 80000 nM T33754 CQWL18 10852535 IC50 > 200000 nM T33754 CCM2Y6 10853678 IC50 = 39000 nM T33754 CE3H7M 10861002 IC50 > 3162.28 nM T33754 CPI5E6 10861494 IC50 < 10000 nM T33754 C8T5KN 10864434 IC50 > 10000 nM T33754 CCV4L0 10873945 IC50 > 3162.28 nM T33754 C3T4WD 10874925 IC50 = 1258.93 nM T33754 C17SLU 10875758 IC50 > 10000 nM T33754 C2DMI8 10885725 IC50 > 10000 nM T33754 CHV5Q1 10885756 IC50 > 10000 nM T33754 CNG12D 10893436 IC50 > 3162.28 nM T33754 CR2I7H 10895319 IC50 > 3162.28 nM T33754 CE4O8T 10896876 IC50 > 3162.28 nM T33754 CRJ5T9 10897006 IC50 > 3162.28 nM T33754 C0RTU9 10897531 IC50 > 10000 nM T33754 CW5EQ0 10903429 IC50 < 10000 nM T33754 C42XNF 10917977 IC50 > 3162.28 nM T33754 C8TJ5Z 10929587 IC50 > 10000 nM T33754 C5UY2I 10940665 IC50 = 794.33 nM T33754 C7W9ZV 10940912 IC50 > 10000 nM T33754 C78BLJ 10962385 IC50 > 10000 nM T33754 CKI1O9 10971811 IC50 > 3162.28 nM T33754 CE1MC0 10980260 IC50 = 5011.87 nM T33754 C58LJN 10981074 IC50 > 3162.28 nM T33754 CR1Y2H 10989584 IC50 = 430 nM T33754 C64POJ 10993740 IC50 > 3162.28 nM T33754 C1R4NH 11004936 IC50 > 3162.28 nM T33754 CE5B8M 11006448 IC50 > 10000 nM T33754 C3AC7X 11015442 IC50 > 3162.28 nM T33754 C3L7EA 11017154 IC50 > 10000 nM T33754 CR7C1N 11017676 IC50 > 10000 nM T33754 CBMN25 11028101 IC50 = 4400 nM T33754 CKBT82 11038706 IC50 > 10000 nM T33754 CIOS65 11038955 IC50 > 10000 nM T33754 CCY7A3 11048935 IC50 > 3162.28 nM T33754 CAD3C4 11050210 IC50 > 10000 nM T33754 C54VZQ 11064194 IC50 = 540 nM T33754 CQI5O1 11067303 IC50 < 10000 nM T33754 CE28QV 11071990 IC50 > 3162.28 nM T33754 CL0VC4 11072016 IC50 > 3162.28 nM T33754 CGW6K3 11072194 IC50 > 10000 nM T33754 CA34RC 11075802 IC50 = 251.19 nM T33754 CX68HJ 11078960 IC50 > 3162.28 nM T33754 C0T1DG 11079584 IC50 > 3162.28 nM T33754 CI2TS9 11079673 IC50 < 10000 nM T33754 CGX54C 11093107 IC50 > 10000 nM T33754 CG74CI 11093245 IC50 > 10000 nM T33754 CT8GE9 11100924 IC50 > 3162.28 nM T33754 C4VJR8 11109680 IC50 < 10000 nM T33754 CG7FV9 11113983 IC50 > 3162.28 nM T33754 CAHJ81 11114030 IC50 > 10000 nM T33754 CR1IZ3 11122701 IC50 > 3162.28 nM T33754 C4C0NX 11122848 IC50 > 10000 nM T33754 CU56SF 11124260 IC50 > 10000 nM T33754 CQ4D5W 11124276 IC50 = 1584.89 nM T33754 C4AET8 11124334 IC50 > 10000 nM T33754 COB72U 11124582 IC50 > 10000 nM T33754 C24VFA 11125005 IC50 > 10000 nM T33754 CU7J6M 11128507 IC50 = 8600 nM T33754 C6KC5Y 11135635 IC50 > 10000 nM T33754 C50SRF 11145589 IC50 > 10000 nM T33754 CR6SE0 11146532 IC50 > 10000 nM T33754 CREQ98 11373312 IC50 = 31000 nM T33754 CU9IY2 11414494 IC50 = 2000 nM T33754 C45VZC 11438405 IC50 > 16000 nM T33754 CV2E4Z 11476710 IC50 = 13000 nM T33754 C4ZYH9 11547485 IC50 > 10000 nM T33754 CKJP43 11723241 IC50 = 35000 nM T33754 CNL0G1 11725859 IC50 > 3000 nM T33754 C1A0KG 11726102 IC50 = 100000 nM T33754 CLR4X2 11729202 IC50 > 3162.28 nM T33754 C2BQ9K 11729404 IC50 < 10000 nM T33754 CX3FQ5 11730938 IC50 > 10000 nM T33754 CB60VT 11733770 IC50 > 10000 nM T33754 C0AKJ4 11742456 IC50 = 12000 nM T33754 CX8J5U 11742876 IC50 > 100000 nM T33754 CFE7S1 11762426 IC50 > 3162.28 nM T33754 CJQ0N8 11775824 IC50 = 170 nM T33754 CK9C5E 11777068 IC50 = 6100 nM T33754 CY0M4H 11777232 IC50 = 140 nM T33754 CQ8Y6L 11793138 IC50 = 30000 nM T33754 CGA1F8 11794425 IC50 = 1000 nM T33754 CYX91E 11795941 IC50 = 40800 nM T33754 C7E8QN 11796403 IC50 = 11000 nM T33754 CYZS05 11798266 IC50 = 19400 nM T33754 C2SXZ1 11798380 IC50 = 19500 nM T33754 C30UGZ 11800567 IC50 > 100000 nM T33754 CBDF71 11812295 IC50 = 8500 nM T33754 CT94GH 11826581 IC50 = 3981.07 nM T33754 C1PM0R 11827787 IC50 > 10000 nM T33754 C29HOL 11828590 IC50 = 8400 nM T33754 CK2J5S 11834125 IC50 > 3162.28 nM T33754 CO9I0H 12016984 IC50 = 48000 nM T33754 CZAV59 12016985 IC50 = 67000 nM T33754 CZ4QA8 12016986 IC50 = 10000 nM T33754 C08RSO 12016987 IC50 = 86000 nM T33754 C4YOB9 12016988 IC50 = 31000 nM T33754 C0VW2U 12016989 IC50 > 100000 nM T33754 C9ZWE6 12016990 IC50 = 120000 nM T33754 C8UL5M 12016991 IC50 = 25000 nM T33754 C28HJD 12016992 IC50 > 100000 nM T33754 CCL4W3 12016993 IC50 = 26000 nM T33754 CAB5E1 12016994 IC50 > 200000 nM T33754 CYF3K5 12016995 IC50 = 102000 nM T33754 CPZ7M4 12726304 IC50 = 100000 nM T33754 C08YKT 12774626 IC50 = 630 nM T33754 CX1CN7 12789009 IC50 = 38000 nM T33754 CP4C7R 12799333 IC50 = 31000 nM T33754 C5RDG7 12850742 IC50 = 1300 nM T33754 COE42X 12851329 IC50 = 2500 nM T33754 CBA94E 12873360 IC50 = 12000 nM T33754 CA5K9I 13037186 IC50 = 16000 nM T33754 CN0UA5 13037188 IC50 = 7300 nM T33754 CE41YR 13059432 IC50 = 7200 nM T33754 CEY1B7 13066339 Ki = 270000 nM T33754 CV79BW 13195776 IC50 = 3400 nM T33754 CNW9B8 13200334 IC50 = 1350 nM T33754 CN9KG3 13232050 IC50 = 40 nM T33754 C7SPV8 13233881 IC50 = 110000 nM T33754 C75JTV 13233882 IC50 = 43000 nM T33754 C9NR8P 13233885 IC50 = 74000 nM T33754 C4AK6E 13233889 IC50 = 2300 nM T33754 CBG9R7 13365079 IC50 = 100000 nM T33754 C15QXF 13365081 IC50 = 43000 nM T33754 CD9SX6 13365089 IC50 = 22000 nM T33754 CJZ8O6 13457698 IC50 = 48 nM T33754 C89SUK 13475879 IC50 = 12100 nM T33754 C1DY8H 13475880 IC50 = 38000 nM T33754 CLU3V4 13475882 IC50 = 160000 nM T33754 C4RK3T 13518856 IC50 = 52000 nM T33754 CRD08J 13518862 IC50 = 22000 nM T33754 CA18FX 13518865 IC50 = 3200 nM T33754 C6G1RO 13535424 IC50 = 400 nM T33754 CPO2I4 13553473 IC50 = 128000 nM T33754 C58VQR 13553476 IC50 = 75000 nM T33754 CN7D9Q 13560740 IC50 = 140 nM T33754 CUT8O7 13560741 IC50 = 140 nM T33754 CN5HR4 13563538 IC50 = 300000 nM T33754 C4LJK9 13563540 IC50 = 38000 nM T33754 C3OHW1 13656051 IC50 = 1800 nM T33754 C6OG1D 13656060 IC50 = 1200 nM T33754 CZRM51 13656069 IC50 = 1600 nM T33754 CH60ZY 13724739 IC50 = 35000 nM T33754 CA35BS 13745706 IC50 = 21000 nM T33754 CL14GZ 13756656 IC50 = 1150 nM T33754 CTZU64 13756657 IC50 = 4400 nM T33754 CU5Z7B 13756658 IC50 = 3600 nM T33754 CRL4Q3 13756663 IC50 = 1300 nM T33754 CL2DO6 13756665 IC50 = 1150 nM T33754 CFKW29 13756666 IC50 = 190 nM T33754 CJXW08 13756670 IC50 = 1800 nM T33754 C6EHB3 13756788 IC50 = 15000 nM T33754 C83QIN 13756791 IC50 = 27000 nM T33754 CD7P5R 13756811 IC50 = 500 nM T33754 C8I5PH 13756813 IC50 = 76000 nM T33754 CX5RB2 13756814 IC50 = 9600 nM T33754 C8SC6J 13813706 IC50 = 129000 nM T33754 C38OTH 13813707 IC50 = 190000 nM T33754 CLO0R8 13813708 IC50 = 25000 nM T33754 CB01QR 13813709 IC50 = 18000 nM T33754 CM25BT 13813714 IC50 = 13000 nM T33754 C1HCW0 13813715 IC50 = 14000 nM T33754 CH4R1T 13854249 IC50 = 870 nM T33754 CZ50CU 13887375 IC50 = 12000 nM T33754 CJWO46 13936973 IC50 = 80 nM T33754 C2W4ML 13936978 IC50 = 20 nM T33754 CI35CU 13936979 IC50 = 35 nM T33754 CT25ZJ 13936981 IC50 = 5 nM T33754 C5M2SC 13936982 IC50 = 8 nM T33754 C0ML2S 13936983 IC50 = 2000 nM T33754 CL9KE4 13936986 IC50 = 3000 nM T33754 CB28RL 13936987 IC50 = 3000 nM T33754 C70FKI 13946679 IC50 = 140000 nM T33754 C6FY4D 13946680 IC50 = 270000 nM T33754 CXE30O 13946684 IC50 = 120000 nM T33754 C9YAU8 13946685 IC50 = 54000 nM T33754 CF49KS 13946687 IC50 = 220000 nM T33754 CF03CE 13946690 IC50 = 590000 nM T33754 CZIR61 13987616 IC50 = 30 nM T33754 CB6DA7 13987617 IC50 = 50 nM T33754 CI9Z6F 13987618 IC50 = 70 nM T33754 C8UVR7 13987619 IC50 = 20 nM T33754 CWYX95 13987620 IC50 = 300 nM T33754 CT05NR 13987621 IC50 = 20 nM T33754 CD6C1Y 13987622 IC50 = 700 nM T33754 CZ7P2Q 13987623 IC50 = 600 nM T33754 CXMG34 13987624 IC50 = 300 nM T33754 CZ6H9F 13987625 IC50 = 5000 nM T33754 C9I1NU 13987626 IC50 = 300 nM T33754 C0HDT3 14067773 IC50 = 7000 nM T33754 CB21VK 14067774 IC50 = 62000 nM T33754 CH4LJ0 14067800 IC50 = 80000 nM T33754 CTK34P 14067801 IC50 = 37000 nM T33754 CV46DH 14067807 IC50 = 5000 nM T33754 CB3N8M 14067808 IC50 = 2000 nM T33754 CJF0S2 14067809 IC50 = 10000 nM T33754 CKI45Q 14067812 IC50 = 128000 nM T33754 C5RJ9F 14067813 IC50 = 2000 nM T33754 CYZ85N 14067814 IC50 = 35000 nM T33754 CASB70 14099426 IC50 = 4100 nM T33754 CI3J7R 14099427 IC50 = 1200 nM T33754 CQ1LY8 14099432 IC50 = 1100 nM T33754 CUS17I 14099444 IC50 = 40000 nM T33754 CP5JU9 14099446 IC50 = 50000 nM T33754 C17HNR 14099449 IC50 = 22000 nM T33754 CZ0YA7 14116989 IC50 = 10000 nM T33754 C8P9XB 14177142 IC50 = 250000 nM T33754 CMF30H 14208192 IC50 > 100000 nM T33754 C85PQM 14230055 IC50 = 9500 nM T33754 C6K8HM 14230056 IC50 = 100000 nM T33754 CCP14U 14230060 IC50 = 100 nM T33754 C0KBQ4 14230061 IC50 = 1000 nM T33754 CH4S8D 14280990 IC50 = 5 nM T33754 CD1Q4U 14280991 IC50 = 600 nM T33754 C03ZNU 14280992 IC50 = 70 nM T33754 CZ9WG1 14280994 IC50 = 5 nM T33754 CL4AF3 14280995 IC50 = 80 nM T33754 C1MK5R 14280996 IC50 = 7000 nM T33754 CCTP04 14280998 IC50 = 30 nM T33754 CXH95F 14280999 IC50 = 5000 nM T33754 CZ6N0W 14281000 IC50 = 40 nM T33754 CR1G8Y 14281001 IC50 = 1 nM T33754 C18OUM 14281003 IC50 = 20 nM T33754 CJ6VF1 14281004 IC50 = 700 nM T33754 CH1BM2 14281005 IC50 = 10 nM T33754 C9MY5X 14281006 IC50 = 0.5 nM T33754 CUCR03 14281008 IC50 = 30 nM T33754 CUFJ35 14281010 IC50 = 100 nM T33754 CQ8TE3 14281011 IC50 = 20 nM T33754 CSEC89 14281012 IC50 = 2000 nM T33754 C85BRF 14281014 IC50 = 2 nM T33754 CU0J8E 14281015 IC50 = 5 nM T33754 CDP92K 14281016 IC50 = 2 nM T33754 C6FCS9 14281018 IC50 = 200 nM T33754 CK3E1F 14281020 IC50 = 80 nM T33754 CUDO17 14281023 IC50 = 500 nM T33754 CZ19AJ 14281024 IC50 = 600 nM T33754 CY8PC6 14281025 IC50 = 2 nM T33754 CBT8K9 14281026 IC50 = 0.4 nM T33754 C3F7MZ 14281027 IC50 = 4 nM T33754 C2CF9I 14281031 IC50 = 50 nM T33754 CQ2YL0 14281033 IC50 = 9 nM T33754 CM1NW7 14281034 IC50 = 100 nM T33754 CEUF73 14281035 IC50 = 30 nM T33754 C7QJ4Y 14281036 IC50 = 300 nM T33754 CWSR46 14281041 IC50 = 100 nM T33754 C69RCW 14373260 IC50 = 40000 nM T33754 CE7L8R 14373269 IC50 = 6400 nM T33754 CB41NR 14373278 IC50 = 14000 nM T33754 C2ZX8H 14756622 IC50 = 300 nM T33754 CIK71M 14836119 IC50 = 15800 nM T33754 CU4B0C 14875705 IC50 = 4000 nM T33754 C0HM4P 14875707 IC50 = 6000 nM T33754 CQE6R7 14978533 IC50 = 9800 nM T33754 CZRD06 14978534 IC50 = 2000 nM T33754 CZ1ML0 15005564 IC50 = 20 nM T33754 CTL89M 15005565 IC50 = 300 nM T33754 CRO7P1 15005566 IC50 = 2000 nM T33754 CCO0S1 15005567 IC50 = 60 nM T33754 C74EYG 15005568 IC50 = 40000 nM T33754 C7RC1U 15005569 IC50 = 1000 nM T33754 CAC98D 15005570 IC50 = 4000 nM T33754 CW0UP4 15005571 IC50 = 4 nM T33754 C6I0LA 15005572 IC50 = 100 nM T33754 CM63ZU 15005573 IC50 = 5000 nM T33754 CE0DR4 15005574 IC50 = 3 nM T33754 CAQ7J2 15005576 IC50 = 2 nM T33754 CTE39J 15005577 IC50 = 0.3 nM T33754 C8TQ6C 15005578 IC50 = 20 nM T33754 C5Z8QA 15005579 IC50 = 8 nM T33754 CS17FZ 15005580 IC50 = 7 nM T33754 CN13YK 15005581 IC50 = 40 nM T33754 CQ9Y7J 15005583 IC50 = 40 nM T33754 CJ72ZA 15005584 IC50 = 20 nM T33754 CVA9B0 15005585 IC50 = 6 nM T33754 C4PM2K 15005586 IC50 = 20 nM T33754 C95NSJ 15005588 IC50 = 6 nM T33754 CI60HD 15005590 IC50 = 3 nM T33754 CDHV05 15005591 IC50 = 100 nM T33754 C7VR0Q 15005592 IC50 = 10 nM T33754 C7QZO0 15005594 IC50 = 2 nM T33754 CP6DI1 15005600 IC50 = 60 nM T33754 C0Z6GL 15005601 IC50 = 100 nM T33754 CTU06K 15005602 IC50 = 600 nM T33754 C23MUZ 15005603 IC50 = 900 nM T33754 CRA5G0 15005604 IC50 = 20 nM T33754 C96YTU 15005605 IC50 = 40 nM T33754 CH7I9M 15005606 IC50 = 300 nM T33754 CX9L6N 15005608 IC50 = 60 nM T33754 C2WC6S 15005610 IC50 = 0.3 nM T33754 C1TUZ8 15005611 IC50 = 7 nM T33754 CK2XC5 15005612 IC50 = 1 nM T33754 CC38GH 15005613 IC50 = 1 nM T33754 C1BWP3 15005614 IC50 = 0.4 nM T33754 C8UXF9 15005615 IC50 = 0.5 nM T33754 CU3OZ1 15005616 IC50 = 0.2 nM T33754 C6FG5L 15005617 IC50 = 0.7 nM T33754 CT7S5U 15005618 IC50 = 0.9 nM T33754 CSB54R 15005619 IC50 = 0.2 nM T33754 CL0GK4 15005620 IC50 = 7 nM T33754 CI9JG7 15005621 IC50 = 0.7 nM T33754 C2PG6E 15005622 IC50 = 2 nM T33754 COXV89 15005623 IC50 = 2 nM T33754 C0RXK5 15005624 IC50 = 9 nM T33754 CLOD12 15005625 IC50 = 0.4 nM T33754 C0NL5Y 15005626 IC50 = 3 nM T33754 CS3BZ0 15005627 IC50 = 0.9 nM T33754 C8RW7L 15005628 IC50 = 2 nM T33754 C5Z1VO 15005629 IC50 = 0.3 nM T33754 C6YWR9 15005630 IC50 = 0.7 nM T33754 C43TXQ 15005631 IC50 = 0.7 nM T33754 CWS8B1 15005632 IC50 = 3 nM T33754 C6MJL0 15005633 IC50 = 0.3 nM T33754 CX2V6D 15005634 IC50 = 0.03 nM T33754 C9PB2Q 15005635 IC50 = 0.6 nM T33754 C3XVH7 15005636 IC50 = 0.08 nM T33754 C5VFK8 15005637 IC50 = 7 nM T33754 C4BJ8X 15005638 IC50 = 5 nM T33754 CU6D4I 15005639 IC50 = 2 nM T33754 CIX0K1 15005640 IC50 = 6 nM T33754 COD9P3 15005641 IC50 = 0.6 nM T33754 CEY94T 15005642 IC50 = 40 nM T33754 CK7IF9 15005643 IC50 = 80 nM T33754 C2FJA7 15005644 IC50 = 30 nM T33754 CAL8G6 15005645 IC50 = 5 nM T33754 CV4N2T 15005646 IC50 = 0.7 nM T33754 CR02FE 15005648 IC50 = 40 nM T33754 C7XTH5 15005649 IC50 = 4 nM T33754 C71XNS 15005650 IC50 = 20 nM T33754 C2FN1U 15005651 IC50 = 40 nM T33754 C4AOZ5 15005652 IC50 = 4.5 nM T33754 C29CGS 15065141 IC50 = 200 nM T33754 CU8Q4O 15065142 IC50 = 300 nM T33754 C6GL1N 15065144 IC50 = 2000 nM T33754 C7FSN1 15065145 IC50 = 50 nM T33754 CI0BC3 15065146 IC50 = 5 nM T33754 CJ9G4E 15065157 IC50 = 150 nM T33754 CJI8S1 15065158 IC50 = 40 nM T33754 C0X4QW 15065159 IC50 = 20000 nM T33754 CDS3L9 15065160 IC50 = 7000 nM T33754 CJAW97 15065161 IC50 = 1500 nM T33754 C6R9QK 15065162 IC50 = 3000 nM T33754 CF2P5L 15065163 IC50 = 3000 nM T33754 C4C9LX 15065166 IC50 = 70000 nM T33754 C1YO3J 15294417 IC50 = 24000 nM T33754 CZ3P9I 15384033 IC50 > 3500 nM T33754 CBI7C9 15599405 IC50 = 50000 nM T33754 C79SKJ 15599407 IC50 = 50000 nM T33754 COIQ39 15599408 IC50 = 100000 nM T33754 C2JFW3 15599410 IC50 = 6000 nM T33754 C9UZY4 15599411 IC50 = 30000 nM T33754 CK85LM 15599412 IC50 = 4000 nM T33754 CL25OI 15599415 IC50 = 630000 nM T33754 CB8AD5 15599416 IC50 = 18000 nM T33754 CKG0I7 15599419 IC50 = 5000 nM T33754 C0FIW4 15599420 IC50 = 6000 nM T33754 CI6PO7 15599423 IC50 = 20000 nM T33754 C9SZV1 15599429 IC50 = 5000 nM T33754 CC7B9I 15599430 IC50 = 8000 nM T33754 CO1B9U 15599431 IC50 = 23000 nM T33754 CZR79K 15599432 IC50 = 36000 nM T33754 CAV9T1 15599433 IC50 = 31000 nM T33754 C7QLW4 15599434 IC50 = 26000 nM T33754 C08RKB 15599435 IC50 = 28000 nM T33754 CF1AI9 15599436 IC50 = 7500 nM T33754 CS62TE 15599439 IC50 = 300 nM T33754 CAC5H0 15606258 IC50 > 100000 nM T33754 C8E9XA 15696722 IC50 = 300 nM T33754 C4ZQ1O 15696723 IC50 = 940 nM T33754 C0ZY9U 15696724 IC50 = 3200 nM T33754 CE50XZ 15717870 IC50 = 2000 nM T33754 CQK95D 15717874 IC50 = 30000 nM T33754 CX4BD2 15717877 IC50 = 7000 nM T33754 CZ4LV6 15717878 IC50 = 45000 nM T33754 C40CME 15717879 IC50 = 40000 nM T33754 CW6MV8 15981426 IC50 = 1300 nM T33754 CL2Y9X 16735134 IC50 = 78 nM T33754 C1PZ8C 18734933 IC50 > 16000 nM T33754 CJ95TM 20146320 IC50 = 3500 nM T33754 CDC76R 20299686 IC50 > 50000 nM T33754 CV74MN 23275981 IC50 = 39810.72 nM T33754 C20VHK 24871823 IC50 = 170 nM T33754 CJ4V0W 44178556 IC50 = 125100 nM T33754 C5X9AD 44209387 IC50 > 100000 nM T33754 C0ZKN1 44209388 IC50 > 100000 nM T33754 CW3O0T 44272155 IC50 = 65000 nM T33754 CNFR26 44272157 IC50 = 10000 nM T33754 CYP61N 44272162 IC50 = 80000 nM T33754 C5ZQN0 44272176 IC50 = 38000 nM T33754 C24ZCG 44272215 IC50 = 40000 nM T33754 CXHP96 44272313 IC50 = 150000 nM T33754 C78OJW 44272327 IC50 = 28000 nM T33754 CSR6M9 44272328 IC50 = 20000 nM T33754 CJ19DZ 44272333 IC50 = 7000 nM T33754 CRO63G 44272338 IC50 = 15000 nM T33754 C1VGQ0 44272341 IC50 = 150000 nM T33754 CRO37P 44274658 IC50 > 100000 nM T33754 C35KNC 44274717 IC50 > 100000 nM T33754 CU36PK 44274868 IC50 > 100000 nM T33754 CDN62V 44274869 IC50 = 840 nM T33754 CA6J8T 44274920 IC50 = 880 nM T33754 CX89AE 44279648 IC50 = 68000 nM T33754 C7NHE8 44279839 IC50 = 220000 nM T33754 CK8Y4F 44286951 IC50 > 50000 nM T33754 CIC45P 44294818 IC50 > 200000 nM T33754 CWTK85 44295026 IC50 > 200000 nM T33754 CEH82G 44295178 IC50 = 250000 nM T33754 CNK73O 44295200 IC50 = 339000 nM T33754 COBW92 44301890 IC50 = 1900 nM T33754 CW75QH 44312546 IC50 = 8 nM T33754 CL80RT 44314758 IC50 = 5300 nM T33754 C3ID9H 44314916 IC50 > 25000 nM T33754 CC6F4N 44315110 IC50 > 100000 nM T33754 C0KT9E 44318468 IC50 < 10000 nM T33754 C4RWG3 44318473 IC50 < 10000 nM T33754 C3L6AF 44319378 IC50 > 3162.28 nM T33754 CLBV45 44320831 IC50 > 10000 nM T33754 CVS5D1 44320863 IC50 > 10000 nM T33754 C0GM7F 44320900 IC50 > 10000 nM T33754 C4VFQ5 44321253 IC50 = 5570 nM T33754 CUQ3R1 44321255 IC50 > 10000 nM T33754 C7BM6I 44321261 IC50 > 10000 nM T33754 CR41FC 44323256 IC50 = 111000 nM T33754 C05VLD 44323257 IC50 = 68000 nM T33754 C2-JAN-01 44323270 IC50 > 200000 nM T33754 CBP5I9 44323409 IC50 > 20000 nM T33754 C0XZ6H 44323410 IC50 > 20000 nM T33754 CK5ZG3 44323424 IC50 > 20000 nM T33754 CFUB24 44323425 IC50 > 20000 nM T33754 CP5N9V 44323427 IC50 > 200000 nM T33754 C5IJQ8 44323428 IC50 > 20000 nM T33754 CMFX02 44323504 IC50 > 20000 nM T33754 C21UJZ 44323510 IC50 = 136000 nM T33754 CAH1Q0 44323556 IC50 > 20000 nM T33754 CTY4U2 44323790 IC50 = 6 nM T33754 CZ16IY 44324251 IC50 = 30000 nM T33754 CCX9Z3 44324252 IC50 = 7000 nM T33754 CG6UT1 44324296 IC50 = 20000 nM T33754 C8M4WJ 44324373 IC50 = 14000 nM T33754 CY5HZ7 44324390 IC50 = 50000 nM T33754 C5KYV6 44324391 IC50 = 50000 nM T33754 C5C4QX 44324507 IC50 = 57000 nM T33754 CXUC09 44329640 IC50 = 430 nM T33754 CA5MY8 44329642 IC50 = 720 nM T33754 CSD45M 44329651 IC50 = 430 nM T33754 CUA7P5 44329666 IC50 = 390 nM T33754 C2M3QE 44329683 IC50 = 310 nM T33754 C9R0OI 44329684 IC50 = 7800 nM T33754 CWM23U 44329685 IC50 = 700 nM T33754 CQ2WU3 44329686 IC50 = 340 nM T33754 CNK2F8 44331802 IC50 = 580 nM T33754 CZ89AS 44333023 IC50 = 10000 nM T33754 CX7E4M 44333357 IC50 = 53000 nM T33754 C5JN7O 44333375 IC50 = 13000 nM T33754 C5ZLT1 44333376 IC50 = 100000 nM T33754 CCOZ32 44339609 IC50 > 300000 nM T33754 C2G4BD 44344410 IC50 = 87000 nM T33754 CA3RE9 44344568 IC50 = 18 nM T33754 CH9P3C 44348937 IC50 = 62000 nM T33754 CVA3O4 44348938 IC50 = 27000 nM T33754 CVW1P2 44348994 IC50 > 100000 nM T33754 C5T6BV 44348995 IC50 = 7850 nM T33754 C2Q9XZ 44349115 IC50 = 17500 nM T33754 C5DKS3 44349135 IC50 = 43700 nM T33754 CS4QH0 44349295 IC50 > 100000 nM T33754 C8L4GH 44350226 IC50 = 200000 nM T33754 CNM4Y5 44350243 IC50 = 4000 nM T33754 C4GDB0 44352576 IC50 > 200000 nM T33754 C0WH4X 44352624 IC50 > 200000 nM T33754 CC3P1L 44352733 IC50 > 200000 nM T33754 C2G1JL 44363503 IC50 = 570 nM T33754 CZX3H7 44364909 IC50 = 5800 nM T33754 C8HWG0 44364924 IC50 = 5400 nM T33754 C9YDX5 44364932 IC50 = 16000 nM T33754 C2WGA3 44365034 IC50 = 11000 nM T33754 CAM5B4 44365046 IC50 = 4800 nM T33754 C9FME0 44365068 IC50 = 125000 nM T33754 CA26VF 44365094 IC50 = 7000 nM T33754 CE0MT4 44365229 IC50 = 6800 nM T33754 C6EBY9 44367306 IC50 > 500000 nM T33754 C7MI2E 44367386 IC50 = 73 nM T33754 CT8NH9 44383851 IC50 > 10000 nM T33754 C19CRH 44383901 IC50 = 3900 nM T33754 CR9O3I 44383902 IC50 = 1100 nM T33754 CW47HV 44383906 IC50 = 2500 nM T33754 CL86MY 44383907 IC50 > 1000 nM T33754 CW63HQ 44383912 IC50 > 1000 nM T33754 CF98LG 44384286 IC50 = 6400 nM T33754 CN1WS7 44384345 IC50 > 10000 nM T33754 C01XPL 44384404 IC50 = 2100 nM T33754 CWPR87 44384405 IC50 = 2100 nM T33754 C59SDR 44384406 IC50 = 3500 nM T33754 C7WT4G 44384540 IC50 = 4500 nM T33754 C4RQB0 44384541 IC50 = 2300 nM T33754 CRZ5G8 44384546 IC50 = 14400 nM T33754 C6W4GY 44384713 IC50 = 8500 nM T33754 CKH7M8 44384714 IC50 = 3600 nM T33754 C0ZGU6 44385109 IC50 = 1500 nM T33754 CE80VB 44385244 IC50 = 840 nM T33754 CH5GU8 44385282 IC50 = 1200 nM T33754 CL50UE 44385283 IC50 = 4400 nM T33754 CZF29N 44397816 IC50 > 10000 nM T33754 C7RV5Q 44438554 IC50 = 1640 nM T33754 C50ZMB 44438560 IC50 = 3130 nM T33754 CJH70L 44438564 IC50 = 1850 nM T33754 C8F3UO 44562338 IC50 = 31.62 nM T33754 C45ZVC 45258276 IC50 = 1500 nM T33754 C2N9HA 45259270 IC50 = 29000 nM T33754 C10TQI 45259276 IC50 = 700 nM T33754 CBKJ47 45259284 IC50 > 100000 nM T33754 CSX9O6 45259293 IC50 = 690 nM T33754 C31FMT 45260180 IC50 > 200000 nM T33754 CCQ35I 45260248 IC50 > 200000 nM T33754 C4BDC7 45261609 IC50 = 77 nM T33754 CSJZ49 45263853 IC50 = 3500 nM T33754 CVSY51 45263858 IC50 = 16000 nM T33754 C1Y9CW 45263914 IC50 = 5600 nM T33754 C0D2MN 46186792 IC50 = 1240 nM T33754 C0WRO9 46198713 IC50 = 7260 nM T33754 CXG34R 46199487 IC50 > 5000 nM T33754 CAL85J 46199794 IC50 > 10000 nM T33754 CI9EA4 46199799 IC50 > 10000 nM T33754 C26RJV 46200090 IC50 > 10000 nM T33754 C5WND9 46200233 IC50 > 10000 nM T33754 CKIC45 46200238 IC50 > 10000 nM T33754 CS46AE 46200399 IC50 > 10000 nM T33754 C1S3BK 46200706 IC50 > 10000 nM T33754 C4P5QJ 46200709 IC50 > 10000 nM T33754 CV8Y6W 46200711 IC50 > 10000 nM T33754 CK1N4X 46200728 IC50 > 1000 nM T33754 CH9FU8 46200877 IC50 > 1000 nM T33754 CEZ3V4 46200878 IC50 = 2250 nM T33754 CI1F5C 46239840 Ki >= 770 nM T33754 C26XVS 46240044 Ki >= 4793 nM T33754 CE4JU7 46842025 IC50 > 10000 nM T33754 CR8JC2 46842169 IC50 > 10000 nM T33754 CIU98Y 49860585 IC50 = 1.13 nM T33754 CV2B7D 49860590 IC50 = 1.13 nM T33754 C7H8OY 49860597 IC50 = 0.84 nM T33754 CS5T3A 49860598 IC50 = 0.63 nM T33754 CSPT34 49860600 IC50 = 1.03 nM T33754 C9Z2SB 49860605 IC50 = 0.81 nM T33754 C0WIU6 49860618 IC50 = 0.81 nM T33754 CBW18A 49860622 IC50 = 2.78 nM T33754 C4U6IX 49860628 IC50 = 1.25 nM T33754 C4D7IC 49860633 IC50 = 5.14 nM T33754 C4KIL0 49860634 IC50 = 2.56 nM T33754 CKD7N1 49860647 IC50 = 1.11 nM T33754 C3EX0U 49860648 IC50 > 10 nM T33754 CP29YZ 49860650 IC50 = 1.13 nM T33754 CN2K8B 49860655 IC50 = 4.96 nM T33754 CBG3J8 49860656 IC50 = 5.42 nM T33754 CURB28 54587645 IC50 = 10000 nM T33754 C0ZF1L 57328385 IC50 > 25000 nM T33754 C2PJ4N 59271992 IC50 = 1000 nM T33754 C7PB1U 59321218 IC50 = 750 nM T33754 CS32XI 59321284 IC50 > 10000 nM T33754 C23WQA 59321310 IC50 > 10000 nM T33754 CZ6C9L 59321318 IC50 > 10000 nM T33754 C1OHZ0 59321339 IC50 > 5000 nM T33754 C0AFM6 60150358 IC50 > 5000 nM T33754 C6C8RD 66802145 IC50 = 1030 nM T33754 CTJ46X 68594477 IC50 > 1000 nM T33754 C8E0XY 68596001 IC50 > 10000 nM T33754 CJ80VI 68596013 IC50 > 10000 nM T33754 CL2H4T 68596452 IC50 > 10000 nM T33754 C93IHS 68596628 IC50 > 10000 nM T33754 CDZ01B 68596639 IC50 > 1000 nM T33754 C1CD9S 68596902 IC50 > 10000 nM T33754 C7PCW0 68597211 IC50 > 1000 nM T33754 CGJB21 68597401 IC50 > 10000 nM T33754 CHK4S0 68597804 IC50 > 10000 nM T33754 C10TGO 68598825 IC50 > 10000 nM T33754 CCN10Q 70662473 IC50 > 1000 nM T33754 CUA5C6 70682518 IC50 = 1680 nM T33754 CPX6Q3 70684576 IC50 = 7490 nM T33754 C2F1WD 70684577 IC50 = 7300 nM T33754 C6DU3W 70686742 IC50 = 312400 nM T33754 C8F2IH 70686743 IC50 = 128300 nM T33754 CM3OP8 70686796 IC50 > 10000 nM T33754 CHBT91 70686797 IC50 > 1000 nM T33754 CJCW26 70688819 IC50 = 38500 nM T33754 C8RHV0 70688820 IC50 = 2660 nM T33754 CYM94A 70688823 IC50 = 8470 nM T33754 CU4I5V 70690900 IC50 = 172500 nM T33754 CR0BM7 70690901 IC50 = 163500 nM T33754 C4YI0P 70695095 IC50 = 423200 nM T33754 CA01QU 70695096 IC50 = 280700 nM T33754 CQR40F 70697129 IC50 = 172130 nM T33754 CF03DW 90168772 IC50 > 20000 nM T33754 CM6J9K 90168778 IC50 > 20000 nM T33754 CVYK24 118556943 IC50 > 50000 nM T33754 C1QMI8 135401477 IC50 > 500 nM T33754 C17YXR 135406983 IC50 > 500 nM T33754 CMHA51 135407168 IC50 = 240 nM T33754 CP3CL2 135410273 IC50 = 150 nM T33754 CXET38 135418296 IC50 = 240 nM T33754 CNP87H 135433645 IC50 > 100000 nM T33754 CMG81E 135434015 IC50 = 3 nM T33754 C94RVJ 135438569 IC50 > 500 nM T33754 CZJY69 135442775 IC50 > 100000 nM T33754 C0DBS7 135452901 IC50 = 62000 nM T33754 CFKO84 135455980 IC50 > 100000 nM T33754 CR6B9J 135456675 IC50 > 100000 nM T33754 C3MWQ9 135474380 IC50 = 83 nM T33754 CGF5P1 135485711 IC50 = 8800 nM T33754 C7SYV0 135506388 IC50 = 2600 nM T33754 CK6CQ7 135515478 IC50 = 72 nM T33754 CB1QD5 135516730 IC50 = 70 nM T33754 CP71WA 135528334 IC50 > 100000 nM T33754 C8E3OA 135531470 IC50 > 100000 nM T33754 C4ASW0 135544141 IC50 > 500 nM T33754 CK8PF5 135583531 IC50 = 520 nM T33754 C7TM3P 135626217 IC50 = 2.7 nM T33754 CZ06BM 135626238 IC50 = 9.2 nM T33754 C58IVM 135626472 IC50 = 48 nM T33754 COJQ24 135626489 IC50 = 5.9 nM T33754 C1XTH2 135626495 IC50 = 1.3 nM T33754 C7WOJ4 135626500 IC50 = 4.6 nM T33754 CQX8E7 135626515 IC50 = 16 nM T33754 CIE79C 135626519 IC50 > 100000 nM T33754 CX06PV 135626541 IC50 = 26 nM T33754 CA8VZ4 135626546 IC50 = 26 nM T33754 C32DLX 135626547 IC50 = 150 nM T33754 C5MDK4 135626551 IC50 = 1.5 nM T33754 CBMT84 135626563 IC50 = 820 nM T33754 CI3PO1 135626568 IC50 = 690 nM T33754 CH8G2M 135626614 IC50 = 3.6 nM T33754 CP81SR 135626617 IC50 = 2000 nM T33754 CJ10HE 135626618 IC50 = 15 nM T33754 C18BJR 135626635 IC50 = 1600 nM T33754 C62SAO 135626651 IC50 = 12 nM T33754 CFS3I4 135626691 IC50 = 2.2 nM T33754 C9MI0X 135626744 IC50 = 5400 nM T33754 C29FKY 135626784 IC50 = 1.45 nM T33754 C5M9KO 135626813 IC50 = 14 nM T33754 C9WI1F 135626836 IC50 = 3.2 nM T33754 C13OYK 135626842 IC50 = 1 nM T33754 CC5Z2N 135666682 IC50 = 600 nM T33754 C3KUC8 135667658 IC50 = 2000 nM T33754 C9OKL0 135668094 IC50 = 700 nM T33754 C7VBI4 135740146 IC50 > 100 nM T33754 CA5NJ0 135823924 IC50 = 1500 nM T33754 C31VFB 135832642 IC50 > 100000 nM T33754 C76RFB 135838394 IC50 = 3300 nM T33754 CE24WD 135838395 IC50 = 40 nM T33754 CRC0Z9 135838396 IC50 = 240 nM T33754 CZOT04 136000670 IC50 = 18000 nM T33754 C8YU1M 136023817 IC50 = 12.5 nM T33754 CR90MI 136026575 IC50 = 8 nM T33754 CTBR86 136026576 IC50 = 6 nM T33754 C6OU3Z 136034782 IC50 > 500 nM T33754 CO9FA3 136035288 IC50 = 300 nM T33754 C5ZIU7 136056125 IC50 > 100000 nM T33754 C70DJG 136056126 IC50 = 34000 nM T33754 C9Q3BW 136056127 IC50 = 63000 nM T33754 C4U1SF 136056128 IC50 = 47000 nM T33754 CI8E5F 136056129 IC50 = 83000 nM T33754 CH92FZ 136058101 IC50 = 290 nM T33754 CI3Z5D 136058102 IC50 = 560 nM T33754 C8PD0K 136058103 IC50 = 600 nM T33754 C13XWR 136058104 IC50 = 26000 nM T33754 CDKT63 136058105 IC50 = 30000 nM T33754 CK8AO5 136058106 IC50 = 18000 nM T33754 CXYS73 136058107 IC50 = 330000 nM T33754 CL42GB 136058108 IC50 = 1500 nM T33754 C6WH2S 136078534 IC50 > 500 nM T33754 C3H7CG 136142433 IC50 = 10000 nM T33754 C4HDJ6 136142434 IC50 > 10000 nM T33754 CUAJ91 136142435 IC50 = 370 nM T33754 CI2K9X 136142436 IC50 = 5.4 nM T33754 C6GH2D 136142437 IC50 = 3300 nM T33754 CU7KY1 136142438 IC50 = 25000 nM T33754 CD2XA8 136142439 IC50 = 17 nM T33754 CLUH17 136142440 IC50 = 1200 nM T33754 CL6CQ7 136142441 IC50 = 27.5 nM T33754 C4O7AN 136142442 IC50 = 4400 nM T33754 CGV71R 136142443 IC50 = 200 nM T33754 CU5OW3 136142444 IC50 = 3800 nM T33754 C45RMB 136142445 IC50 = 1000 nM T33754 CSMY91 136142446 IC50 > 10000 nM T33754 CI5W0G 136142447 IC50 = 6.4 nM T33754 CR7V3M 136142448 IC50 > 10000 nM T33754 C9KH1P 136142449 IC50 = 6 nM T33754 C4Y1QU 136142450 IC50 = 580 nM T33754 C5NPS9 136142451 IC50 = 26 nM T33754 CIN5D2 136142452 IC50 = 340 nM T33754 C7WPY3 136142453 IC50 = 4.1 nM T33754 CEW57J 136142454 IC50 = 1 nM T33754 CIH0D9 136142455 IC50 = 1600 nM T33754 CID97M 136142456 IC50 = 4.9 nM T33754 CH2U9V 136142457 IC50 = 260 nM T33754 CTM6W3 136142458 IC50 = 1600 nM T33754 C8TGF9 136142459 IC50 = 18.5 nM T33754 CMNO98 136142460 IC50 = 1.85 nM T33754 CO34ZP 136142461 IC50 = 76 nM T33754 C7VJX6 136142462 IC50 = 5 nM T33754 C7HG8U 136142463 IC50 = 5.6 nM T33754 CMO62W 136142464 IC50 = 13.5 nM T33754 CTZR90 136142465 IC50 = 180 nM T33754 CYR1K6 136142466 IC50 = 11 nM T33754 COS9I7 136142467 IC50 = 2 nM T33754 C4VW9B 136142468 IC50 = 120 nM T33754 CND42L 136142469 IC50 = 12 nM T33754 CXZM43 136142470 IC50 = 1.1 nM T33754 C9S8RE 136142471 IC50 = 1.45 nM T33754 C8EVA1 136142472 IC50 = 18 nM T33754 CY49SD 136142473 IC50 = 10 nM T33754 C0J9IZ 136142474 IC50 = 0.94 nM T33754 C1QHS2 136142476 IC50 = 760 nM T33754 C0EV7C 136142477 IC50 = 4.5 nM T33754 CIP98Q 136142478 IC50 = 3100 nM T33754 CY9EB3 136142479 IC50 = 1700 nM T33754 C2VI5E 136142480 IC50 = 470 nM T33754 CD9IK1 136142481 IC50 = 130 nM T33754 CA6BF0 136142482 IC50 = 140 nM T33754 C6CZW9 136144096 IC50 = 13 nM T33754 CQW7T0 136197286 IC50 > 10000 nM T33754 D00YPO 14032753 IC50 = 110 nM T33754 D01RUN 448055 IC50 > 3162.28 nM T33754 D01TOR 667555 IC50 > 100000 nM T33754 D02NWF 2573787 IC50 > 100000 nM T33754 D03GAQ 15065156 IC50 = 10 nM T33754 D04KDB 13885278 IC50 = 16000 nM T33754 D05HFD 13936971 IC50 = 50 nM T33754 D08XKO 15065155 IC50 = 300 nM T33754 D09AUL 10266864 IC50 = 50000 nM T33754 D09CPC 13728862 IC50 = 4400 nM T33754 D09GTN 13936969 IC50 = 300 nM T33754 D09LAQ 135398570 IC50 = 2400 nM T33754 D0DL6J 9843744 IC50 > 100000 nM T33754 D0DX3V 13936989 IC50 = 20 nM T33754 D0I6XA 149784 Ki > 200000 nM T33754 D0J0CB 2753 Ki = 5 nM T33754 D0J7GF 780643 IC50 > 100000 nM T33754 D0J7NR 15065143 IC50 = 90 nM T33754 D0LZ5R 5368 IC50 > 100000 nM T33754 D0N6MR 10867033 IC50 = 500 nM T33754 D0NI4Z 13936972 IC50 = 50 nM T33754 D0O3BL 19700663 IC50 = 5100 nM T33754 D0S4JI 20262 IC50 > 200000 nM T33754 D0T3UP 13724742 IC50 = 7000 nM T33754 D0TZ8C 14373279 IC50 = 4000 nM T33754 D0U8YQ 921562 IC50 > 100000 nM T33754 D0V4WB 149790 IC50 > 16000 nM T33754 D0V5BX 68765 IC50 > 200000 nM T95947 D0I0RJ 16231 IC50 = 4400 nM T95947 CV9U4J 237074 IC50 = 97000 nM T95947 C98HYW 350414 IC50 = 363000 nM T95947 CWQ6T8 598430 IC50 = 763000 nM T95947 CF8D7P 817383 IC50 = 130000 nM T95947 C2L8DB 910176 IC50 = 430000 nM T95947 C5DZ4S 2762833 IC50 = 6900 nM T95947 C1FXO2 3010990 IC50 = 6300 nM T95947 CJ79MR 11160454 IC50 = 9000 nM T95947 C4HR0W 11413259 IC50 = 190000 nM T95947 C0OKV6 15885183 IC50 = 701000 nM T95947 C9JO6S 21473659 IC50 = 3300 nM T95947 CEG0S4 25210286 IC50 = 133000 nM T95947 CL8F3J 25254508 IC50 = 95000 nM T95947 CN1A2U 25254510 IC50 = 374000 nM T95947 CVJ09D 25254512 IC50 = 77000 nM T95947 CGP5U4 29949062 IC50 = 160000 nM T95947 CQG62F 42630453 IC50 = 490 nM T95947 CNB07T 44276630 IC50 = 2765000 nM T95947 CIRV37 44574852 IC50 = 510 nM T95947 C3UZ1O 44575053 IC50 = 640 nM T95947 CA13UC 45268405 IC50 = 135000 nM T95947 CUD7O4 45268406 IC50 = 278000 nM T95947 CBY5A2 45270104 IC50 = 291000 nM T95947 C2UM9J 45270105 IC50 = 59000 nM T95947 CGVY53 45270945 IC50 = 114000 nM T95947 CK36FD 45272657 IC50 = 272000 nM T95947 CRT7U8 45272658 IC50 = 59000 nM T95947 CH4P7Z 45273577 IC50 = 51000 nM T95947 CT3F0N 53235532 IC50 = 3800 nM T95947 CG69CQ 53327817 IC50 = 3100 nM T95947 CC5JU4 53357591 IC50 = 220 nM T95947 CV8O9S 54580851 IC50 = 10900 nM T95947 C8DU2L 54580852 IC50 = 1700 nM T95947 CL2VD1 54581911 IC50 = 27600 nM T95947 C6JNA1 54581912 IC50 = 7100 nM T95947 C7FXW8 54581913 IC50 = 103000 nM T95947 CMR50V 54582827 IC50 = 17000 nM T95947 C2CWP3 54582828 IC50 = 9600 nM T95947 CM2N0V 54583845 IC50 = 14400 nM T95947 CVH03X 54585747 IC50 = 5800 nM T95947 CF93ML 54586726 IC50 = 19400 nM T95947 C5J3IG 54587763 IC50 = 2600 nM T95947 C8I7BE 54587764 IC50 = 1200 nM T95947 CXD10Y 56659437 IC50 > 50000 nM T95947 CZE85N 56659438 IC50 > 50000 nM T95947 CG0D5O 56659439 IC50 = 2500 nM T95947 C4PVI5 56662841 IC50 = 17100 nM T95947 C3VU5T 56662880 IC50 = 460 nM T95947 C8S0UA 56662881 IC50 = 4800 nM T95947 C5PC6Y 56662884 IC50 = 510 nM T95947 CK18MS 56666368 IC50 = 230 nM T95947 CDTA43 56666369 IC50 = 10200 nM T95947 C7UCQ9 56669778 IC50 = 310 nM T95947 C4Y2VS 56669779 IC50 = 230 nM T95947 C29ZIH 56669780 IC50 = 190 nM T95947 CX65FU 56673271 IC50 = 2800 nM T95947 COB8C7 56676588 IC50 = 270 nM T95947 CLT4K0 56679936 IC50 = 680 nM T95947 C5JMB3 56683256 IC50 = 3400 nM T95947 CSG38B 56683258 IC50 = 4300 nM T25315 D00XBC 46861584 IC50 > 10000 nM T25315 CLK7P3 169713 IC50 > 10000 nM T25315 C8TI6Z 197750 IC50 = 4570 nM T25315 CQX4M9 265219 IC50 > 60000 nM T25315 CEV5K8 384454 IC50 > 100000 nM T25315 CXQE10 384455 IC50 = 8000 nM T25315 C80QFG 384457 IC50 = 3000 nM T25315 CK20TD 594995 IC50 = 800 nM T25315 C3KCR4 703047 IC50 = 800 nM T25315 CB3Y5H 703050 IC50 = 3500 nM T25315 CLC86X 742729 IC50 = 4000 nM T25315 CX3FU4 871434 IC50 = 1100 nM T25315 CCAR78 1378429 Ki = 3981.07 nM T25315 CX6VK4 1448380 IC50 > 12589.25 nM T25315 CK6BI3 2396278 IC50 = 2940 nM T25315 COT07B 3453336 IC50 > 60000 nM T25315 C85BVJ 4239764 Ki = 3981.07 nM T25315 CG2MN3 4324393 IC50 = 250 nM T25315 CJB37A 6143230 Ki = 211 nM T25315 C86QRZ 9871365 IC50 = 3300 nM T25315 C1ZF0K 9886775 Ki = 110 nM T25315 C2PM8U 9913494 IC50 = 15000 nM T25315 CUB3G7 9938326 IC50 = 6 nM T25315 CMUB67 9938965 IC50 = 14 nM T25315 C81TFE 11296495 IC50 = 20 nM T25315 C97LDW 11386761 IC50 = 930 nM T25315 CVGK31 11497512 Ki = 140 nM T25315 C8TX6O 11498089 IC50 = 11 nM T25315 C1Y6EO 11526863 Ki = 160 nM T25315 CMGN54 11569938 IC50 = 0.2 nM T25315 CR0Q7V 11599725 IC50 = 35 nM T25315 CLQ14F 11635543 Ki = 320 nM T25315 CMZ08A 11707105 Ki = 85 nM T25315 C39SQF 11713886 Ki = 70 nM T25315 CWA39Z 11725848 IC50 = 2000 nM T25315 CNPX34 11757854 IC50 = 4.1 nM T25315 C91ZWK 11854699 IC50 = 6.8 nM T25315 C5EN9M 11856829 IC50 = 1.3 nM T25315 CE5AL8 11856830 IC50 = 1.4 nM T25315 CB8X2P 11964007 IC50 = 8 nM T25315 CJ1V6Z 11995700 IC50 = 1 nM T25315 C0P3HV 11995702 IC50 = 1.2 nM T25315 C7ZXA5 11995703 IC50 = 1.3 nM T25315 CYP1D7 11995772 IC50 = 9 nM T25315 CM71UD 11995774 Ki = 0.4 nM T25315 C2SR7I 11995974 IC50 = 2 nM T25315 C6B2LT 11995976 IC50 = 2.2 nM T25315 C8YLS5 11996050 IC50 = 1.5 nM T25315 C2VO4N 11996051 IC50 = 1.9 nM T25315 C1OM3A 11996344 IC50 = 1.9 nM T25315 C96NUB 11996409 IC50 = 3.9 nM T25315 C3J1YV 11996560 IC50 = 4.2 nM T25315 CZQ47C 11996722 IC50 = 5.2 nM T25315 C9PY6Q 11996726 IC50 = 6 nM T25315 C3FV2N 11997121 IC50 = 5.4 nM T25315 CD8P4G 11997270 IC50 = 18 nM T25315 CH6S5Q 11997334 IC50 = 1.8 nM T25315 CWR74C 11997336 IC50 = 6.4 nM T25315 CXSV02 11997474 IC50 = 3.6 nM T25315 CX0BJ7 11997620 IC50 = 1.5 nM T25315 CFQE74 11997623 IC50 = 3.4 nM T25315 CW6DT4 11997695 IC50 = 0.3 nM T25315 CD2WH3 11997761 IC50 = 0.4 nM T25315 CH21MR 11997845 IC50 = 0.4 nM T25315 CW0OT8 11997912 IC50 = 0.8 nM T25315 CRF9W1 11997994 IC50 = 0.8 nM T25315 C56KLN 11997995 IC50 = 0.3 nM T25315 C3DAP8 14479861 IC50 = 830 nM T25315 C19BYU 14479864 IC50 = 330 nM T25315 CNOH94 15560447 IC50 = 2400 nM T25315 C4C1BL 15604604 IC50 = 60 nM T25315 CY8QA1 15604606 IC50 = 120 nM T25315 CD4XZ9 15604607 IC50 = 170 nM T25315 C8AYG5 15604608 IC50 = 1250 nM T25315 CA3F2D 15604688 IC50 = 700 nM T25315 CJWO23 15604689 IC50 = 130 nM T25315 C80SEI 15604690 IC50 = 800 nM T25315 C9X7KF 15604773 IC50 = 80 nM T25315 CQD8K4 15604774 IC50 = 300 nM T25315 C65NQZ 15604776 IC50 = 2160 nM T25315 CYB49S 15604856 IC50 = 60 nM T25315 CZC28M 15604859 IC50 = 340 nM T25315 CF37DQ 15604934 IC50 = 320 nM T25315 C5GCE0 15604935 IC50 = 60 nM T25315 CL5ZI0 15604937 IC50 = 420 nM T25315 CT0B6H 15604938 IC50 = 240 nM T25315 CD3U7V 15605007 IC50 = 590 nM T25315 CSM0E4 15605012 IC50 = 490 nM T25315 CI4F5R 15605071 IC50 = 340 nM T25315 CF2RE4 15605073 IC50 = 250 nM T25315 CPIL45 15605074 IC50 = 50 nM T25315 C2O6LA 15605075 IC50 = 510 nM T25315 CUC1O6 15605137 IC50 = 290 nM T25315 CE29DR 15605197 IC50 = 70 nM T25315 CC1FM8 15605618 IC50 = 640 nM T25315 CV3NQ0 16040696 IC50 = 11 nM T25315 C2ARS4 16214851 IC50 = 3162.28 nM T25315 CX32OZ 17754430 IC50 = 2200 nM T25315 C97IHN 17754488 IC50 = 30 nM T25315 C8NYG4 17754713 IC50 = 800 nM T25315 C6C4QK 17754758 IC50 = 400 nM T25315 CX18AK 17754794 IC50 = 8000 nM T25315 CJI3V4 17754798 IC50 = 800 nM T25315 CAQ7S0 17754836 IC50 = 1000 nM T25315 C1CG7D 23593653 IC50 = 3100 nM T25315 CETZ25 23790139 IC50 = 40000 nM T25315 C7N4BG 24739386 IC50 = 150 nM T25315 C8KTP0 24739387 IC50 = 2310 nM T25315 CN9SZ0 24739388 IC50 = 210 nM T25315 C70CVK 24739554 IC50 = 30 nM T25315 C7K5DU 24739555 IC50 = 320 nM T25315 CSDA50 24739886 IC50 = 80 nM T25315 C12LWD 24739888 IC50 = 290 nM T25315 CY09OP 24739889 IC50 = 250 nM T25315 CMPR25 24774715 IC50 = 340 nM T25315 CUY89J 24936155 Ki = 7 nM T25315 CYLZ53 24947459 IC50 = 794.33 nM T25315 C0V8YL 24957182 IC50 = 8 nM T25315 C7D6KF 25008271 IC50 = 80 nM T25315 COH9V1 25032696 IC50 = 12 nM T25315 C9E6YT 25032697 IC50 = 7.8 nM T25315 C5NE1L 25032779 IC50 = 2 nM T25315 CJ32HC 25265835 IC50 = 31.62 nM T25315 C5NZI8 27307547 IC50 = 251.19 nM T25315 CAE5J4 34747495 IC50 = 2275 nM T25315 C5O1MR 44137674 IC50 = 7 nM T25315 C5ZJG2 44138054 Ki = 158.49 nM T25315 CYN7W6 44182602 IC50 = 7 nM T25315 C4E0DK 44237762 IC50 = 25 nM T25315 C5YFB9 44252324 IC50 > 10000 nM T25315 C31VGY 44253167 IC50 = 1295 nM T25315 C4H6BG 44253168 IC50 = 200 nM T25315 CV17CB 44253169 IC50 = 1985 nM T25315 C6P4LJ 44253170 IC50 = 2450 nM T25315 C42OMV 44253446 IC50 = 496 nM T25315 CYU6I9 44253447 IC50 = 697 nM T25315 C8C0YJ 44253448 IC50 = 673 nM T25315 CX3H2E 44253449 IC50 = 695 nM T25315 CC1IH2 44253450 IC50 = 470 nM T25315 CZ1OH8 44253589 IC50 = 1295 nM T25315 CM5F3V 44253590 IC50 = 2560 nM T25315 C1P2EV 44253591 IC50 = 1460 nM T25315 C0CQV9 44253592 IC50 = 885 nM T25315 CZ5Y7Q 44253594 IC50 = 5580 nM T25315 C4R6FA 44253725 IC50 = 940 nM T25315 CR6AY7 44253726 IC50 = 510 nM T25315 C28BEU 44253727 IC50 = 347 nM T25315 CWO8B6 44402370 IC50 = 10000 nM T25315 CPRD27 44402504 IC50 > 100000 nM T25315 C13SIY 44402582 IC50 = 5800 nM T25315 C8QL3D 44402658 IC50 > 100000 nM T25315 CTE82I 44406196 IC50 = 200 nM T25315 C8S4YD 44406244 IC50 = 890 nM T25315 C1CND2 44406261 IC50 = 3100 nM T25315 CVHX75 44406274 IC50 = 250 nM T25315 C7M4TS 44406319 IC50 = 190 nM T25315 CEK68R 44406343 IC50 = 9800 nM T25315 CC7P8K 44406348 IC50 = 13000 nM T25315 CQDI02 44406362 IC50 = 2150 nM T25315 CYWF12 44426595 IC50 = 146 nM T25315 C8E7FG 44426596 IC50 > 10000 nM T25315 C8VG5B 44426676 IC50 = 154 nM T25315 CE25ZP 44426677 IC50 = 375 nM T25315 CJM9Y8 44426678 IC50 > 10000 nM T25315 CU1QV3 44426679 IC50 = 710 nM T25315 CG9F8V 44426680 IC50 = 790 nM T25315 C3USK7 44426681 IC50 = 587 nM T25315 CQF50T 44426682 IC50 = 1400 nM T25315 CNQK92 44426684 IC50 = 75 nM T25315 CA4WI1 44426685 IC50 > 10000 nM T25315 CQ59ES 44426687 IC50 > 10000 nM T25315 CE8KT6 44426689 IC50 > 10000 nM T25315 C10DNL 44426690 IC50 = 88 nM T25315 CU2I9R 44426691 IC50 = 156 nM T25315 CD02AO 44426693 IC50 = 300 nM T25315 CQPA38 44426694 IC50 = 40 nM T25315 CW7QO3 44426696 IC50 > 10000 nM T25315 C39YWG 44426697 IC50 = 100 nM T25315 C1IB7A 44426698 IC50 = 230 nM T25315 CC3HX1 44426700 IC50 = 650 nM T25315 CHX5L4 44426702 IC50 = 240 nM T25315 CAYN63 44426704 IC50 = 73 nM T25315 CX59SN 44426705 IC50 = 12 nM T25315 CZP36J 44426707 IC50 = 299 nM T25315 C2XM8V 44426709 IC50 = 22 nM T25315 C8MTK3 44426710 IC50 = 25 nM T25315 CS26WG 44426711 IC50 = 14 nM T25315 C3JGN9 44426712 IC50 = 4 nM T25315 CI9VE2 44426713 IC50 = 7 nM T25315 C1IVP3 44426714 IC50 = 11 nM T25315 CAN3Z0 44426715 IC50 = 10000 nM T25315 CM36CB 44426716 IC50 = 1370 nM T25315 CWG81F 44426717 IC50 = 25000 nM T25315 CF8TQ5 44426718 IC50 = 2300 nM T25315 C9PC4S 44426719 IC50 = 75 nM T25315 CP1W5K 44426720 IC50 > 10000 nM T25315 C1VS2L 44426721 IC50 = 9 nM T25315 C7CAD8 44426722 IC50 = 4000 nM T25315 C2PW9U 44426723 IC50 = 6 nM T25315 CMD9W8 44426724 IC50 = 144 nM T25315 CQN23M 44426725 IC50 = 1400 nM T25315 C3YVD8 44426726 IC50 = 480 nM T25315 CZ1HM8 44426909 Ki = 88 nM T25315 CX6JZ7 44426911 Ki = 201 nM T25315 CCR8I3 44426912 Ki = 104 nM T25315 C1YA3J 44426913 Ki = 637 nM T25315 CF5T6J 44426914 Ki = 36 nM T25315 CYG30D 44426915 Ki = 47 nM T25315 C7B5KO 44426917 Ki = 41 nM T25315 CY0QL7 44426920 Ki = 306 nM T25315 CSQ39F 44426931 Ki = 1040 nM T25315 C92KYE 44426932 Ki = 3400 nM T25315 C8HXV6 44426934 Ki = 660 nM T25315 C6EPQ5 44426935 Ki = 108 nM T25315 C10HDQ 44426990 Ki = 290 nM T25315 C9NPB6 44426992 Ki = 1300 nM T25315 C56CNU 44426993 Ki = 2200 nM T25315 C9HBE6 44426994 Ki = 2000 nM T25315 C7G6VX 44426995 Ki = 26 nM T25315 C5TCJ4 44426996 Ki = 258 nM T25315 CJ52DF 44426998 Ki = 171 nM T25315 C62OEC 44426999 Ki = 429 nM T25315 C8FME2 44427000 Ki = 31 nM T25315 CZG57H 44427001 Ki = 175 nM T25315 CH41ZJ 44427002 Ki = 191 nM T25315 C6PA3B 44427003 Ki = 39 nM T25315 CWLV83 44427004 Ki = 29 nM T25315 C8QVY7 44427005 Ki = 46 nM T25315 CPGI84 44427006 Ki = 171 nM T25315 C2NPL3 44427007 Ki = 70 nM T25315 CE4U2C 44427008 Ki = 107 nM T25315 CB57WJ 44427009 Ki = 141 nM T25315 C1DQ9J 44427010 Ki = 83 nM T25315 CXE68Z 44427011 Ki = 191 nM T25315 CKCI49 44427013 Ki = 229 nM T25315 CQM6I9 44427014 Ki = 16 nM T25315 CG58XD 44427015 Ki = 81 nM T25315 C26PAQ 44427016 Ki = 376 nM T25315 CRK03J 44427019 Ki = 28 nM T25315 COI4D1 44443757 Ki = 180 nM T25315 CJ2X4L 44443759 Ki = 3600 nM T25315 CY1CM8 44443799 Ki = 3500 nM T25315 CT3AG0 44443812 Ki = 170 nM T25315 C06FOM 44443813 Ki = 200 nM T25315 CCI0V1 44443814 Ki = 680 nM T25315 CC0BL6 44443816 Ki = 720 nM T25315 CDG70K 44443818 Ki = 350 nM T25315 CUKG03 44443820 Ki = 126 nM T25315 C7N8FP 44443821 Ki = 950 nM T25315 C8M6OE 44443822 Ki = 460 nM T25315 CC5BH3 44443823 Ki = 290 nM T25315 CG06SI 44443825 Ki = 170 nM T25315 C7QU8A 44443827 Ki = 620 nM T25315 CR16SG 44443828 Ki = 150 nM T25315 CF58ZA 44443830 Ki = 130 nM T25315 C5GN2J 44443831 Ki = 880 nM T25315 CFR4S3 44443833 Ki = 460 nM T25315 CMZ3F8 44443834 Ki = 260 nM T25315 C8VTC4 44443835 Ki = 270 nM T25315 CXFA79 44446421 Ki = 1100 nM T25315 CKEW28 44446422 Ki = 180 nM T25315 C19WRK 44446423 Ki = 60 nM T25315 C6PR0N 44446438 Ki = 190 nM T25315 C41QLD 44446439 Ki = 27 nM T25315 CPH8N9 44446441 Ki = 28 nM T25315 C2JBE3 44446443 Ki = 20 nM T25315 C0HWP6 44446445 Ki = 18 nM T25315 C8C4IX 44446450 Ki = 9 nM T25315 CK6DR1 44446451 Ki = 10 nM T25315 CRG6O5 44446452 Ki = 280 nM T25315 C5CZ1N 44446453 Ki = 11 nM T25315 CTPF78 44446454 Ki = 3 nM T25315 CV4Q3Z 44446457 Ki = 120 nM T25315 CT27ON 44447090 IC50 = 21 nM T25315 CMS98X 44447091 IC50 = 27 nM T25315 CU5TN2 44447092 IC50 = 9 nM T25315 CCV03Y 44447093 IC50 = 5 nM T25315 CCZ7G4 44447094 IC50 = 4 nM T25315 CZ41CV 44447095 IC50 = 35 nM T25315 C45PYZ 44447096 Ki = 3 nM T25315 CV13QK 44447097 IC50 = 10 nM T25315 CY9ZH4 44447098 IC50 = 523 nM T25315 C2CM7R 44453168 IC50 = 15 nM T25315 CHC2Z8 44453201 IC50 = 400 nM T25315 CJ9MS5 44453232 IC50 = 100 nM T25315 CP2K3T 44453266 IC50 = 400 nM T25315 C67XKC 44453267 IC50 = 300 nM T25315 C74BMH 44453295 IC50 = 2300 nM T25315 C6OT8Y 44453296 IC50 = 800 nM T25315 CURJ65 44453322 IC50 = 500 nM T25315 CHP8R7 44453362 IC50 = 3400 nM T25315 CI8KQ3 44453364 IC50 = 200 nM T25315 CFNV87 44453439 IC50 = 1200 nM T25315 CP59RA 44453468 IC50 = 20 nM T25315 C4G1XC 44453470 IC50 = 20 nM T25315 C7VRC2 44453530 IC50 = 16 nM T25315 CCN36G 44453558 IC50 = 15 nM T25315 C3HLJ5 44453583 IC50 = 15 nM T25315 CW6M5E 44453585 IC50 = 20 nM T25315 CGC18I 44453616 IC50 = 20 nM T25315 CX24TY 44453640 IC50 = 20 nM T25315 C43LJW 44453643 IC50 = 20 nM T25315 CVAR89 44454490 IC50 = 11000 nM T25315 CD39AJ 44454491 IC50 = 22000 nM T25315 C68PRZ 44454492 IC50 = 3000 nM T25315 CQ15UF 44454527 IC50 = 16000 nM T25315 CR02BQ 44454588 IC50 = 20000 nM T25315 CLV09T 44454589 IC50 = 50000 nM T25315 CW28RB 44454591 IC50 = 11000 nM T25315 CR36OC 44454616 IC50 > 50000 nM T25315 CR7S1T 44454617 IC50 > 50000 nM T25315 CL6X9V 44454618 IC50 > 50000 nM T25315 CI06HS 44454619 IC50 > 50000 nM T25315 C8MYB0 44454644 IC50 = 3000 nM T25315 CD7HP9 44454645 IC50 > 100000 nM T25315 CS2RV7 44454796 IC50 = 700 nM T25315 CF0HE2 44454824 IC50 = 400 nM T25315 CRZ0S7 44454826 IC50 = 300 nM T25315 C9AM2E 44454895 IC50 = 5000 nM T25315 CTDO37 44454934 IC50 = 6000 nM T25315 CHMX10 44455463 IC50 = 10 nM T25315 CS07AT 44455464 IC50 = 8 nM T25315 C4B8RZ 44455480 Ki = 6 nM T25315 CDP34N 44455488 IC50 = 3.8 nM T25315 CAMQ81 44455489 IC50 = 3.2 nM T25315 CN63DX 44455507 Ki = 5 nM T25315 C0WGY8 44455508 Ki = 4 nM T25315 CLO97I 44455517 IC50 = 2.5 nM T25315 CQ2U0J 44455536 Ki = 3 nM T25315 C63XVT 44455537 Ki = 6 nM T25315 C9SHN8 44455538 Ki = 24 nM T25315 CQO4A5 44455542 IC50 = 2.6 nM T25315 C4AUD2 44455558 Ki = 25 nM T25315 CJL93M 44455559 Ki = 20 nM T25315 CGN9O2 44455561 Ki = 7 nM T25315 CO9M7F 44455565 IC50 = 6.6 nM T25315 C3LA2F 44455568 IC50 = 29 nM T25315 C7LH6V 44455569 IC50 = 43 nM T25315 C8FNQ3 44455591 Ki = 18 nM T25315 C6L5HC 44455592 Ki = 21 nM T25315 C85IXV 44455593 Ki = 26 nM T25315 CD9JS4 44455603 IC50 = 40 nM T25315 C4RM3X 44455604 IC50 = 0.7 nM T25315 C3Z8RN 44455621 Ki = 624 nM T25315 C1JY6K 44455623 Ki = 15 nM T25315 C0AT4Q 44455624 Ki = 143 nM T25315 C7AF4M 44455634 IC50 = 44 nM T25315 CK9CF3 44455640 IC50 = 2.1 nM T25315 CD7R2O 44455656 Ki = 95 nM T25315 CGA1N7 44455657 Ki = 135 nM T25315 CK3P0E 44455668 IC50 = 9.4 nM T25315 CF1MA0 44455669 IC50 = 5 nM T25315 CYK1C0 44455693 IC50 = 5.6 nM T25315 C8SJ1R 44455722 IC50 = 7.1 nM T25315 CT5LU2 44455723 IC50 = 4.8 nM T25315 CM83TF 44455751 IC50 = 0.4 nM T25315 C6YB5X 44455752 IC50 = 2.4 nM T25315 C3ER7Q 44455773 IC50 = 6.4 nM T25315 CJ85LG 44455774 IC50 = 11 nM T25315 C07RWG 44455799 IC50 = 36 nM T25315 CD7A6G 44455800 IC50 = 11 nM T25315 CE8IV9 44455801 IC50 = 81 nM T25315 CR0PD3 44455823 IC50 = 129 nM T25315 CTKJ17 44455824 IC50 = 1179 nM T25315 C4U8KC 44455825 IC50 = 752 nM T25315 CVMQ03 44455843 IC50 = 1.8 nM T25315 CY5X1B 44455852 IC50 = 72 nM T25315 CC73TZ 44455870 IC50 = 3 nM T25315 CE0J4D 44455873 IC50 = 19 nM T25315 C67ECQ 44569941 IC50 = 1584.89 nM T25315 C50RXU 44569942 IC50 = 158.49 nM T25315 CIF8H1 44569943 IC50 = 794.33 nM T25315 C7O6MC 44569944 IC50 = 199.53 nM T25315 CA9FG7 44570029 IC50 = 199.53 nM T25315 CPG92E 44570140 IC50 = 794.33 nM T25315 C9JL0W 44570141 IC50 = 1995.26 nM T25315 CPY61G 44570142 IC50 = 630.96 nM T25315 CFI5O3 44570178 IC50 = 794.33 nM T25315 CB52AH 44570179 IC50 = 7943.28 nM T25315 CWLT20 44570180 IC50 = 79.43 nM T25315 C8MJK1 44570181 IC50 = 501.19 nM T25315 CGCZ05 44570218 IC50 = 316.23 nM T25315 C5Y0GJ 44570219 IC50 = 158.49 nM T25315 C9NED2 44570220 IC50 = 31.62 nM T25315 CA6W4U 44570221 IC50 = 316.23 nM T25315 CZJ2Y0 44570272 IC50 = 50.12 nM T25315 C6P5BJ 44570273 IC50 = 63.1 nM T25315 C12LRN 44570274 IC50 = 39.81 nM T25315 C1JI8N 44570310 IC50 > 31622.78 nM T25315 CH41VM 44570311 IC50 = 25118.86 nM T25315 C6JL8T 44570312 IC50 = 125.89 nM T25315 CE3D5K 44570340 IC50 = 25118.86 nM T25315 CG3L8N 44570341 IC50 = 1584.89 nM T25315 C3R9CO 44570342 IC50 > 31622.78 nM T25315 CV1K2L 44570343 IC50 > 31622.78 nM T25315 CKMS98 44570344 IC50 > 31622.78 nM T25315 CK2I7F 44570383 IC50 > 31622.78 nM T25315 CJ1Y4O 44570384 IC50 > 31622.78 nM T25315 C06TEU 44570385 IC50 = 158.49 nM T25315 CGI97J 44570430 IC50 = 398.11 nM T25315 CT59OX 44570431 IC50 = 251.19 nM T25315 C7Q4LA 44570432 IC50 = 316.23 nM T25315 CQL02F 44570433 IC50 > 31622.78 nM T25315 CA1JV3 44570470 IC50 = 1995.26 nM T25315 CSZN78 44570471 IC50 = 316.23 nM T25315 CXC47F 44570472 IC50 = 630.96 nM T25315 C2SBW1 44570473 IC50 = 5011.87 nM T25315 CSZ10Q 44570515 IC50 = 15848.93 nM T25315 CK7MT9 44570516 IC50 = 316.23 nM T25315 C9YJ5C 44570517 IC50 = 630.96 nM T25315 C6EM9O 44570547 IC50 = 6309.57 nM T25315 CT92VI 44570548 IC50 > 31622.78 nM T25315 CSA37U 44570549 IC50 = 158.49 nM T25315 CBK73R 44570550 IC50 = 501.19 nM T25315 CXH83L 44570595 IC50 = 398.11 nM T25315 CQ47MB 44570596 IC50 = 630.96 nM T25315 CGH57K 44570597 IC50 > 31622.78 nM T25315 C3WNP8 44570598 IC50 > 31622.78 nM T25315 CHEF64 44570627 IC50 = 6309.57 nM T25315 CZY82W 44570628 IC50 = 31622.78 nM T25315 CD81NC 44570629 IC50 = 15848.93 nM T25315 CR1EN7 44570630 IC50 > 31622.78 nM T25315 CFMI18 44580796 IC50 = 790 nM T25315 CW7C5I 44580797 IC50 = 1260 nM T25315 C80DQT 44580798 IC50 = 320 nM T25315 C0KC9I 44580799 IC50 = 1000 nM T25315 CH2NB1 44580823 IC50 = 2510 nM T25315 CFRD71 44580857 IC50 = 2510 nM T25315 CW8DX0 44580858 IC50 = 5010 nM T25315 CA7T9E 44580859 IC50 = 5010 nM T25315 CQ64PE 44580860 IC50 = 2000 nM T25315 CEI7X4 44580878 IC50 = 1000 nM T25315 C6VZX1 44580902 IC50 = 690 nM T25315 CAD63V 44580903 IC50 = 180 nM T25315 CTS8M1 44580939 IC50 = 500 nM T25315 C7ZI2N 44580959 IC50 > 10000 nM T25315 C7JDB3 44580960 IC50 = 1580 nM T25315 CM5FR3 44581069 IC50 = 4270 nM T25315 CX6ZC8 44581070 IC50 = 3160 nM T25315 C27TFX 44581087 IC50 = 1260 nM T25315 CM08HC 44581088 IC50 = 2510 nM T25315 CBDG70 44581089 IC50 = 500 nM T25315 CSGK97 44581090 IC50 = 1000 nM T25315 CJP27F 44581108 IC50 = 630 nM T25315 C0PRS3 44581109 IC50 = 1260 nM T25315 CF13RW 44581110 IC50 = 3630 nM T25315 CS92ZI 44581134 IC50 = 1550 nM T25315 C2YCI0 44581135 IC50 = 170 nM T25315 COXU45 44581136 IC50 = 1450 nM T25315 C3S7LY 44581137 IC50 = 5010 nM T25315 CO7CH6 44581159 IC50 = 630 nM T25315 CR04AU 44581160 IC50 = 3160 nM T25315 CTQG38 44581161 IC50 = 3160 nM T25315 C52KSR 44581162 IC50 = 1260 nM T25315 CK68GB 44591872 Ki = 501.19 nM T25315 CH83XO 44591873 Ki = 501.19 nM T25315 C3BZ1U 44591874 Ki = 6309.57 nM T25315 CQ68TX 44591875 Ki > 10000 nM T25315 CM3CL2 44591885 Ki = 6309.57 nM T25315 CWBE05 44591886 Ki = 3981.07 nM T25315 CFI43D 44591887 Ki = 1584.89 nM T25315 CJ4CW7 44591918 Ki = 794.33 nM T25315 CYLA46 44591928 Ki = 1258.93 nM T25315 C63BCT 44592137 IC50 = 0.3 nM T25315 C8ZGH3 44592138 Ki > 100000 nM T25315 CSX5I3 44592139 Ki = 5011.87 nM T25315 CHEZ19 44592140 Ki > 10000 nM T25315 C0P3TB 44592174 Ki = 2511.89 nM T25315 C8I0QU 44592175 Ki = 5011.87 nM T25315 CL43NG 44592176 Ki = 3981.07 nM T25315 C0V1OK 44592177 Ki = 3981.07 nM T25315 CNQY29 44592178 Ki > 10000 nM T25315 CXB0Y1 44592220 Ki = 398.11 nM T25315 C6ET4R 44592221 Ki = 1000 nM T25315 CM5P7L 44592222 Ki = 1000 nM T25315 C5A1PQ 44592264 Ki = 501.19 nM T25315 CS7H3P 44592265 Ki = 1258.93 nM T25315 C3RS7M 44592266 Ki = 2511.89 nM T25315 CTXG85 44592267 Ki = 501.19 nM T25315 C0YIB3 44592268 Ki = 7943.28 nM T25315 CY8V9H 44592304 Ki = 5011.87 nM T25315 CNS17G 44592305 Ki = 3981.07 nM T25315 C0CKI4 44592306 Ki = 5011.87 nM T25315 CG5FQ2 44592341 Ki = 3981.07 nM T25315 CYS8Z3 44592342 Ki = 1995.26 nM T25315 C8P4HM 44592343 Ki = 1584.89 nM T25315 C80SLH 44592344 Ki > 10000 nM T25315 CUYP04 44592403 Ki = 3162.28 nM T25315 CI6CP5 44592404 Ki = 794.33 nM T25315 CXM01D 44592405 Ki = 10000 nM T25315 C1TO8P 44592406 Ki = 7943.28 nM T25315 CL9F5P 44592407 Ki = 1995.26 nM T25315 C1G6UJ 44592471 Ki = 1584.89 nM T25315 CGH7F5 44592472 Ki = 1995.26 nM T25315 C1OBI0 44592473 Ki = 398.11 nM T25315 CV0NE9 44592474 Ki = 2511.89 nM T25315 CO9U6M 44592475 Ki = 7943.28 nM T25315 CNCT24 44592527 Ki > 10000 nM T25315 CV4ZX1 44592528 Ki = 6309.57 nM T25315 C0T6OI 44592529 Ki = 2511.89 nM T25315 CT0B1I 44592530 Ki = 3981.07 nM T25315 CIR39K 44592531 Ki = 1995.26 nM T25315 CNZ1U7 44593651 IC50 = 60 nM T25315 C7DK9G 44593733 Ki = 398.11 nM T25315 C5JGD4 44593735 Ki = 3981.07 nM T25315 CSHE04 45101497 IC50 = 16 nM T25315 C3P5FJ 45101498 IC50 = 32 nM T25315 CM6C9Q 45101529 IC50 = 0.4 nM T25315 C9HZ2R 45379650 IC50 = 0.9 nM T25315 C8A1FM 45482784 IC50 = 179 nM T25315 C0CHF4 45482789 IC50 = 18 nM T25315 CG09IA 45482794 IC50 > 10000 nM T25315 CA7MT2 45482795 IC50 = 231 nM T25315 CU07RG 45482796 IC50 = 803 nM T25315 CS7H4A 45482800 IC50 = 2000 nM T25315 CTO70Z 45482803 IC50 > 10000 nM T25315 CK0NU7 45482807 IC50 = 100 nM T25315 C07UTP 45482808 IC50 = 564 nM T25315 CNK31C 45482813 IC50 > 10000 nM T25315 CEP68M 45482814 IC50 = 1930 nM T25315 C82CZS 45482819 IC50 = 62 nM T25315 C92SGJ 45482823 IC50 = 67 nM T25315 CUH5N1 45482836 IC50 = 60 nM T25315 CCN71E 45482843 IC50 = 510 nM T25315 CVT85J 45482849 IC50 = 28 nM T25315 C1E7BH 45484653 Ki = 870 nM T25315 C6GUW2 45484655 Ki = 1900 nM T25315 CZ19CS 45484656 IC50 = 560 nM T25315 CCV7W8 45484657 Ki = 3700 nM T25315 C95ONL 45484658 Ki = 90 nM T25315 C1EZ5R 45484671 Ki = 370 nM T25315 CX1Q9P 45484678 Ki = 4100 nM T25315 CPR4Y6 45484679 Ki = 470 nM T25315 CEK34W 45484680 Ki = 3800 nM T25315 CTX6G2 45484691 Ki = 510 nM T25315 C2WA8F 45484692 Ki = 330 nM T25315 CNEQ82 45484705 Ki = 410 nM T25315 CT1NL4 45484716 Ki = 8900 nM T25315 CXB16P 45484733 Ki = 1900 nM T25315 CR6Y2Q 45484739 IC50 = 20 nM T25315 CBMG60 45484740 Ki > 50000 nM T25315 CZ4YW9 45484748 Ki = 120 nM T25315 CA95WT 45484749 Ki = 2900 nM T25315 CBH0R2 45485420 IC50 = 4500 nM T25315 CRFG06 45485423 Ki = 7200 nM T25315 C27GJB 45485429 Ki = 86 nM T25315 CER5O9 45485434 Ki = 16 nM T25315 CB6C0G 45485437 Ki = 32 nM T25315 CO45AX 45485438 Ki = 2000 nM T25315 CH4LC2 45485451 Ki = 2700 nM T25315 CHUM15 45485458 Ki = 23000 nM T25315 CUON70 45486493 IC50 = 2 nM T25315 CGN04B 45486520 IC50 = 60 nM T25315 CCPR31 45486521 IC50 = 3 nM T25315 CM1GD4 45486522 IC50 = 18 nM T25315 CAN49B 45486523 IC50 = 0.9 nM T25315 C5CG6H 45486524 IC50 = 1.6 nM T25315 CVB49D 45486525 IC50 = 1.1 nM T25315 CL49VY 45486526 IC50 = 0.9 nM T25315 CSW98R 45486528 IC50 = 1.4 nM T25315 CSB01J 45486529 IC50 = 44 nM T25315 CEHV82 45486530 IC50 = 1.1 nM T25315 CX8JN5 45486531 IC50 = 21 nM T25315 C6DVW7 45486532 IC50 = 29 nM T25315 C1YZT7 45486533 IC50 = 1.3 nM T25315 C9SDX2 45486534 IC50 = 1.1 nM T25315 CVD09X 45486555 IC50 = 4 nM T25315 C0B1JF 45486556 IC50 = 4 nM T25315 C4A5KL 45486557 IC50 = 457 nM T25315 C9UZS8 45486558 IC50 > 1000 nM T25315 C93HDC 45486559 IC50 = 29 nM T25315 C69LTY 45486560 IC50 = 10 nM T25315 CT3V4F 45486561 IC50 = 3 nM T25315 CK8QW4 46225413 IC50 > 60000 nM T25315 C92GWM 46700871 IC50 = 192 nM T25315 CP57KH 46883287 IC50 = 690 nM T25315 C5UM7W 46883288 IC50 = 210 nM T25315 CLS3E6 46883289 IC50 = 7 nM T25315 CB2M8T 46883290 IC50 = 13 nM T25315 C9IL1T 46883291 IC50 = 2090 nM T25315 CKWP14 46883292 IC50 = 11 nM T25315 CRK72O 46883293 IC50 = 21 nM T25315 CRX7I9 46883294 IC50 = 770 nM T25315 CA2L3W 46883295 IC50 = 40 nM T25315 CT56QR 46883296 IC50 = 8 nM T25315 CT1XY7 46883297 IC50 = 7 nM T25315 C0P2ZK 46883298 IC50 = 9 nM T25315 C3JU1T 46883299 IC50 = 2 nM T25315 CYF17Z 46883300 IC50 = 23 nM T25315 CBJI21 46883301 IC50 = 110 nM T25315 CF29SM 46883302 IC50 = 42 nM T25315 C12RTY 46883303 IC50 = 2 nM T25315 CNU64B 46883304 IC50 = 10 nM T25315 CPH4U2 46883305 IC50 = 5 nM T25315 C6Y5AE 46883306 IC50 = 2 nM T25315 CBAR75 46883307 IC50 = 2 nM T25315 C61ADL 46883308 IC50 = 1 nM T25315 C8WH2O 46883309 IC50 = 131 nM T25315 C32OKX 46883310 IC50 = 5 nM T25315 C1U2JO 46883311 IC50 = 1 nM T25315 CF1WQ6 46890724 IC50 = 183 nM T25315 CNBY78 46890725 IC50 = 339 nM T25315 C7PRW5 46890726 IC50 = 216 nM T25315 CC80EV 46890727 IC50 = 207 nM T25315 CL9RS8 46891078 IC50 = 192 nM T25315 C8HMI6 46891145 IC50 = 238 nM T25315 C05ZXW 46891183 IC50 = 85 nM T25315 CG4IZ3 46891223 IC50 = 1152 nM T25315 C0RJ7G 46891224 IC50 = 360 nM T25315 C49ELR 46891272 IC50 = 13 nM T25315 C17TKX 46891273 IC50 = 6440 nM T25315 CZ6KG3 46891327 IC50 = 1132 nM T25315 CHXZ61 46891328 IC50 = 513 nM T25315 CYL9S8 46891329 IC50 = 1080 nM T25315 C5WA4D 46891371 IC50 = 882 nM T25315 C70PAG 46891424 IC50 = 233 nM T25315 C8X6IK 46891425 IC50 = 540 nM T25315 CPU40W 46891476 IC50 = 911 nM T25315 C4LNX0 46891477 IC50 = 254 nM T25315 CE7R5I 46891478 IC50 = 440 nM T25315 CM6JR5 46891536 IC50 = 158 nM T25315 COJS83 46891537 IC50 = 157 nM T25315 C2W6HF 46891538 IC50 = 236 nM T25315 C5VHE3 46893277 Ki = 199.53 nM T25315 CQAT71 53317216 IC50 = 8100 nM T25315 CIH6U1 53317274 IC50 = 31 nM T25315 CQ8RT1 53317275 IC50 = 520 nM T25315 C4M8QS 53317276 IC50 = 2.4 nM T25315 C84QKU 53317277 IC50 = 22 nM T25315 CNA91W 53317663 IC50 = 83 nM T25315 CBX25C 53318510 IC50 = 17 nM T25315 CG5R8E 53318511 IC50 > 10000 nM T25315 C0LNA3 53318512 IC50 = 1980 nM T25315 CSN30W 53318513 IC50 = 58 nM T25315 C06OAZ 53318514 IC50 = 210 nM T25315 CDCA26 53318560 IC50 = 6 nM T25315 CYS7N6 53318561 IC50 = 7000 nM T25315 CUM62K 53318562 IC50 = 280 nM T25315 CCF2J7 53318563 IC50 = 8900 nM T25315 C1M5SJ 53318914 IC50 = 830 nM T25315 CV3AR4 53319879 IC50 = 39 nM T25315 CT7KC2 53319880 IC50 = 64 nM T25315 CYP2B1 53319881 IC50 = 20 nM T25315 C68LPB 53319882 IC50 = 32 nM T25315 C6M5QK 53321134 IC50 > 10000 nM T25315 C0OG1S 53321184 IC50 = 39 nM T25315 CO0VP5 53321185 IC50 = 5 nM T25315 C3W9GC 53321186 IC50 = 3100 nM T25315 C5AZ9K 53321187 IC50 = 23 nM T25315 CRAG94 53322459 IC50 = 5 nM T25315 C4F2WR 53322460 IC50 = 63 nM T25315 C17FLG 53322461 IC50 = 8060 nM T25315 CXL54M 53322503 IC50 > 10000 nM T25315 CS37NB 53322504 IC50 = 40 nM T25315 C64WRQ 53322505 IC50 = 2700 nM T25315 CZSY87 53322506 IC50 = 27 nM T25315 C04FJG 53322507 IC50 = 7350 nM T25315 C3VGE4 53322508 IC50 = 8 nM T25315 CHJ16M 53322509 IC50 = 2.3 nM T25315 C13HWL 53322510 IC50 = 900 nM T25315 CPY5A1 53322511 IC50 = 630 nM T25315 CGK9M0 53322974 IC50 = 7990 nM T25315 C7EG5Q 53323853 IC50 = 140 nM T25315 CY2QU7 53323854 IC50 = 910 nM T25315 CF85ZO 53324231 IC50 = 3 nM T25315 C7TL6S 53324328 IC50 > 50000 nM T25315 CZ7B8C 53325131 IC50 = 1400 nM T25315 CYFL35 53325132 IC50 = 12500 nM T25315 CB0ZI6 53325133 IC50 = 80 nM T25315 CST63J 53325134 IC50 = 260 nM T25315 CI90MS 53326388 IC50 = 18 nM T25315 CXFS62 53326389 IC50 = 87 nM T25315 CIWZ65 53326434 IC50 = 220 nM T25315 CI2F1D 53326850 IC50 = 29 nM T25315 CVP7O2 54764847 IC50 = 1.3 nM T25315 C2TF8D 56660098 IC50 = 305 nM T25315 C4IB1X 56660099 IC50 = 12 nM T25315 CXJ5Q0 56660100 IC50 = 81 nM T25315 C3Y4MP 56660101 IC50 = 16 nM T25315 CK7CU3 56660102 IC50 = 5 nM T25315 CXGA53 56663557 IC50 = 17 nM T25315 CE6OU8 56663558 IC50 = 67 nM T25315 CA1MK4 56663559 IC50 = 22 nM T25315 CNM6R8 56663560 IC50 = 3 nM T25315 C9Y7XJ 56663561 IC50 = 53 nM T25315 CGZ58A 56663562 IC50 = 5 nM T25315 C3TF1C 56663563 IC50 = 8 nM T25315 C4EH6A 56667005 IC50 = 457 nM T25315 C7WH3Y 56667006 IC50 = 200 nM T25315 C90ZSJ 56667007 IC50 = 20 nM T25315 C7ZS8I 56667008 IC50 > 10000 nM T25315 C6TX1V 56667009 IC50 = 14 nM T25315 CE5B0W 56670448 IC50 = 14 nM T25315 CZI80K 56670449 IC50 = 12 nM T25315 CHPD72 56670450 IC50 = 523 nM T25315 CRX87E 56670451 IC50 = 27 nM T25315 C6KFM1 56670452 IC50 = 6200 nM T25315 CINM64 56670453 IC50 > 10000 nM T25315 C6NP4T 56670454 IC50 = 2200 nM T25315 CM9QG4 56670455 IC50 = 2600 nM T25315 CU1I9Y 56670456 IC50 = 170 nM T25315 C04IPB 56670465 IC50 = 28 nM T25315 C53OLI 56673431 IC50 = 4 nM T25315 CG7AL2 56673937 IC50 = 9 nM T25315 CSD20W 56673938 IC50 = 83 nM T25315 C68OUR 56673939 IC50 = 216 nM T25315 C13WYF 56673940 IC50 = 7 nM T25315 C7R3CU 56673941 IC50 = 160 nM T25315 C4TA3N 56673942 IC50 = 11 nM T25315 CCZ98M 56673943 IC50 = 9475 nM T25315 CW4J1Y 56673944 IC50 = 2 nM T25315 CKW4Z0 56673945 IC50 = 3 nM T25315 CB0MR9 56673953 IC50 > 10000 nM T25315 CH7NA4 56677270 IC50 = 825 nM T25315 CN58TZ 56677271 IC50 = 4 nM T25315 CDC12H 56677272 IC50 = 89 nM T25315 C4SB5Y 56677273 IC50 = 8 nM T25315 CLW35V 56677274 IC50 = 6120 nM T25315 CYA6W7 56680570 IC50 = 12 nM T25315 CNE8Q0 56680571 IC50 = 74 nM T25315 CM4H9X 56680572 IC50 = 5400 nM T25315 CJ2B3H 56680573 IC50 > 10000 nM T25315 CFU4D9 56680574 IC50 = 5 nM T25315 CWV06G 56680588 IC50 = 379 nM T25315 C7V9WR 56683907 IC50 > 10000 nM T25315 CPN57V 56834986 IC50 = 12 nM T25315 C9B3IZ 57390182 IC50 = 29 nM T25315 C0G9RK 57390209 IC50 = 7 nM T25315 C5NRS1 57390764 IC50 = 2.5 nM T25315 CB5GH2 57390765 IC50 = 0.9 nM T25315 CJ9E8I 57392573 IC50 = 3.7 nM T25315 C2W4QX 57392574 IC50 = 0.9 nM T25315 CVY53H 57392575 IC50 = 2.9 nM T25315 C71AYV 57392576 IC50 > 1000 nM T25315 CXP8A9 57393685 IC50 = 21 nM T25315 C2ZXG7 57394143 IC50 = 8 nM T25315 CA4L9P 57394299 IC50 = 1.5 nM T25315 CFCI01 57394300 IC50 = 1.8 nM T25315 CJ06XR 57394301 IC50 = 1.1 nM T25315 C0CU3Q 57396053 IC50 = 8.4 nM T25315 CZ47JD 57396054 IC50 = 4.4 nM T25315 CIE8P1 57396055 IC50 = 1.9 nM T25315 CIU06Z 57397852 IC50 = 8.5 nM T25315 C4L2BA 57397853 IC50 = 6.4 nM T25315 C80THO 57397854 IC50 = 3.4 nM T25315 CV1T4M 57397855 IC50 = 1.5 nM T25315 C0SMP4 57397856 IC50 = 1.9 nM T25315 C3WMN4 57399515 IC50 = 4 nM T25315 C15KWV 57399516 IC50 = 2.4 nM T25315 C6FIN0 57399517 IC50 = 2 nM T25315 CXNA63 57399518 IC50 = 235 nM T25315 C6WJU5 57400628 IC50 = 47 nM T25315 CRL27H 57400629 IC50 = 6 nM T25315 CB7UI1 57400677 IC50 = 50 nM T25315 CJ6T7Z 57401268 IC50 = 4.1 nM T25315 CVJ60W 57401269 IC50 = 1.2 nM T25315 C1TQ0D 57401270 IC50 = 3.6 nM T25315 CT7HP6 57402420 IC50 = 7 nM T25315 CF74AH 57402421 IC50 = 6 nM T25315 C4Y6LX 57403018 IC50 = 76 nM T25315 C2MOF3 57403019 IC50 = 2.9 nM T25315 CMCR69 57403020 IC50 = 4.2 nM T25315 CFD1H9 58186816 IC50 = 23.6 nM T25315 C0YWT1 58509213 IC50 > 10000 nM T25315 CW9QE3 58767992 IC50 = 33.8 nM T25315 CO9A1X 58768002 IC50 = 24.5 nM T25315 CV4WM6 58768027 IC50 = 1.8 nM T25315 C5AS8M 58768044 IC50 = 3.8 nM T25315 CZ35PK 58768048 IC50 = 1.2 nM T25315 CP8LT7 58768061 IC50 = 1.6 nM T25315 CN8MZ0 58768069 IC50 = 6.2 nM T25315 C2UDL3 59772540 IC50 = 286 nM T25315 CZS67E 59772541 IC50 = 0.3 nM T25315 C7R1OE 59772590 IC50 = 1376 nM T25315 C9TZ1U 68102990 IC50 = 50.5 nM T25315 CF3IV1 71450265 Ki = 50.12 nM T25315 C7H1TE 71450267 Ki = 2511.89 nM T25315 C8JQ5C 71450269 Ki = 158.49 nM T25315 CB6NI2 71450271 Ki = 1000 nM T25315 CN9E6V 71450472 Ki = 251.19 nM T25315 C2MDO0 71450474 Ki = 501.19 nM T25315 C08PIB 71450476 Ki > 316.23 nM T25315 CV94LS 71450477 Ki > 316.23 nM T25315 CYKW92 71450478 Ki > 316.23 nM T25315 C3QDS2 71450479 Ki > 316.23 nM T25315 CMS83A 71450527 Ki > 316.23 nM T25315 CQU7C0 71450528 Ki = 1584.89 nM T25315 CZD30U 71450530 Ki = 1000 nM T25315 C9SEQ1 71450532 Ki = 630.96 nM T25315 CKE64U 71450534 Ki = 630.96 nM T25315 C76YQS 71450536 Ki = 15848.93 nM T25315 CU6F5I 71450537 Ki = 2511.89 nM T25315 C64OBF 71450539 Ki = 3981.07 nM T25315 C20ATU 71450540 Ki = 794.33 nM T25315 CS8D3F 71452091 Ki = 501.19 nM T25315 CZ2LN6 71452093 Ki = 100 nM T25315 C7ASV4 71452310 Ki = 199.53 nM T25315 CF3Z1I 71452312 Ki = 316.23 nM T25315 CWOG46 71452314 Ki = 3981.07 nM T25315 CQ2MD5 71452315 Ki = 1000 nM T25315 CQ3IJ8 71452374 Ki = 3162.28 nM T25315 CC1JU7 71452375 Ki = 1995.26 nM T25315 C4Y5XB 71452377 Ki = 398.11 nM T25315 CFNK04 71452379 Ki = 7943.28 nM T25315 C07AYL 71452380 Ki = 3162.28 nM T25315 C5N6XV 71452381 Ki = 7943.28 nM T25315 CIS53Z 71453923 Ki = 398.11 nM T25315 C4Q3FX 71453925 Ki = 398.11 nM T25315 CBV1L9 71454100 Ki = 199.53 nM T25315 C25LRG 71454102 Ki = 1584.89 nM T25315 C8DQT6 71454104 Ki = 3162.28 nM T25315 C8H6RA 71454154 Ki > 316.23 nM T25315 C2LM8W 71454155 Ki = 2511.89 nM T25315 CCSO26 71454157 Ki = 7943.28 nM T25315 CYM0Z5 71455652 Ki = 158.49 nM T25315 CGLO60 71455654 Ki = 501.19 nM T25315 C5ZY7U 71455656 Ki = 100 nM T25315 CIC9O6 71455658 Ki = 398.11 nM T25315 CY93MX 71455837 Ki = 501.19 nM T25315 CHN98F 71455839 Ki = 3162.28 nM T25315 CV6B5G 71455841 Ki = 2511.89 nM T25315 CBQ85T 71455884 Ki = 1995.26 nM T25315 C3JD5K 71455885 Ki = 251.19 nM T25315 CPL57Q 71455887 Ki = 5011.87 nM T25315 CQK5Y0 71455888 Ki = 12589.25 nM T25315 C4UZH2 71455889 Ki = 3162.28 nM T25315 CNG1V3 71457435 Ki = 199.53 nM T25315 CAG4P3 71457437 Ki = 501.19 nM T25315 CHCE02 71457439 Ki = 39.81 nM T25315 CX58ZE 71457631 Ki = 398.11 nM T25315 CN36SQ 71457633 Ki = 1258.93 nM T25315 C13TZU 71457635 Ki = 6309.57 nM T25315 CP4WI9 71457636 Ki = 6309.57 nM T25315 CKJ27M 71457637 Ki > 316.23 nM T25315 C9GQO8 71457681 Ki = 1258.93 nM T25315 CW8G7L 71457683 Ki > 316.23 nM T25315 C4U0ZV 71457684 Ki = 2511.89 nM T25315 CC6QB3 71457685 Ki = 3162.28 nM T25315 CX1QO7 71459294 Ki = 63.1 nM T25315 CV7H9J 71459296 Ki = 501.19 nM T25315 CESM84 71459298 Ki = 630.96 nM T25315 C9TU4O 71459300 Ki = 199.53 nM T25315 CKM67R 71459302 Ki = 1995.26 nM T25315 CUYV29 71459523 Ki = 501.19 nM T25315 CXFU13 71459525 Ki > 316.23 nM T25315 CF4YM2 71459526 Ki > 316.23 nM T25315 CJ76KX 71459589 Ki = 316.23 nM T25315 C51UFM 71459591 Ki = 1995.26 nM T25315 C1T7DQ 71459593 Ki = 5011.87 nM T25315 C8B5LH 71459594 Ki = 5011.87 nM T25315 CK4AL7 71461073 Ki = 63.1 nM T25315 C5Y6DG 71461075 Ki = 125.89 nM T25315 C86CVJ 71461268 Ki = 630.96 nM T25315 C2ZJN0 71461270 Ki = 501.19 nM T25315 CSE9N6 71461272 Ki > 316.23 nM T25315 CGT2E1 71461273 Ki = 1995.26 nM T25315 CM5U7K 71461327 Ki > 316.23 nM T25315 CERW83 71461328 Ki = 1000 nM T25315 CQ2AS1 71461330 Ki = 1584.89 nM T25315 C3TGQ2 71461332 Ki = 6309.57 nM T25315 CF9K4W 71462809 Ki = 199.53 nM T25315 CM94FX 71462811 Ki = 316.23 nM T25315 CE63CT 71462813 Ki = 316.23 nM T25315 CP35IU 71462815 Ki = 251.19 nM T25315 C3U2YV 71462992 Ki = 1000 nM T25315 CT07HI 71462994 Ki = 398.11 nM T25315 C23LZH 71462996 Ki > 316.23 nM T25315 C6LDC4 71462997 Ki > 316.23 nM T25315 CS5F0N 71462998 Ki = 3981.07 nM T25315 C2ZF9P 71463056 Ki > 316.23 nM T25315 CFZ76K 71463057 Ki = 7943.28 nM T25315 C92XFW 71572192 IC50 = 13 nM T25315 C5D4UG 71585199 IC50 = 76 nM T25315 CT9FC8 71585298 IC50 = 99 nM T25315 CS2F9Z 71585504 IC50 = 1000 nM T25315 CN4TC7 71586201 IC50 = 60 nM T25315 C5J1QB 71586204 IC50 = 19 nM T25315 CG9Q0A 71586301 IC50 = 38 nM T25315 CY07QP 71586303 IC50 = 24 nM T25315 C27AGH 71586392 IC50 = 200 nM T25315 CV41FJ 71586393 IC50 = 37 nM T25315 C01KZL 71586394 IC50 = 35 nM T25315 C7DAX6 71586395 IC50 = 44 nM T25315 C4LZA0 71586485 IC50 = 55 nM T25315 CTIM92 71586679 IC50 = 53 nM T25315 C98ABQ 72188563 IC50 = 11 nM T25315 CNR52H 72547710 IC50 = 424 nM T25315 CEA80B 72547711 IC50 = 74 nM T25315 C5KND0 72547938 IC50 = 71 nM T25315 C5NXI9 72547939 IC50 = 81 nM T25315 C3NMQ1 72548178 IC50 = 81 nM T25315 CZC5F9 72549346 IC50 = 41 nM T25315 C0I7GV 72549347 IC50 = 34 nM T25315 CU49SV 72549349 IC50 = 44 nM T25315 C51ZCM 72549350 IC50 = 23 nM T25315 CP1WC8 72549588 IC50 = 108 nM T25315 CB40JU 72549589 IC50 = 95 nM T25315 C9XVJ7 72549590 IC50 = 677 nM T25315 C6J3EX 72549591 IC50 = 130 nM T25315 CNV52I 72549592 IC50 = 42 nM T25315 CIOM39 72549594 IC50 = 428 nM T25315 CWO36A 72549595 IC50 = 123 nM T25315 CTR8J1 72549596 IC50 = 440 nM T25315 CE4Y9I 72549821 IC50 = 31 nM T25315 CU5CS1 72550475 IC50 = 70 nM T25315 C0UP9J 72550699 IC50 = 143 nM T25315 CS74JL 76317929 IC50 = 437 nM T25315 CL4YU8 76325253 IC50 = 2295 nM T25315 C0EHJ3 76332481 IC50 = 1.6 nM T25315 CYWE71 89610442 IC50 = 1060 nM T25315 C0WE2I 89610499 IC50 = 176 nM T25315 C9QGW5 89610658 IC50 = 23 nM T25315 C7JG5M 89610683 IC50 = 25 nM T25315 CB59GM 89610699 IC50 = 607 nM T25315 CYCF45 89610786 IC50 = 26 nM T25315 CA0Z4U 90014266 IC50 = 61 nM T25315 CZ4L0V 90014377 IC50 = 152 nM T25315 CZ6Y5V 90014385 IC50 = 69 nM T25315 C5JC7Z 90014472 IC50 = 110 nM T25315 CMP3K2 90014508 IC50 = 73 nM T25315 CNB2Y5 90014551 IC50 = 256 nM T25315 CH0I5G 90014572 IC50 = 21 nM T25315 CE8FK0 90014593 IC50 = 263 nM T25315 C7J0VY 90014675 IC50 = 154 nM T25315 C85BYS 90014688 IC50 = 96 nM T25315 C74FIX 90014694 IC50 = 122 nM T25315 C76PCB 90014714 IC50 = 47 nM T25315 CNDX82 90014722 IC50 = 80 nM T25315 CEX71F 90014726 IC50 = 132 nM T25315 C9PD3S 90014869 IC50 = 146 nM T25315 CUV32W 90014874 IC50 = 91 nM T25315 C2YD5H 90015039 IC50 = 118 nM T25315 C24OKV 90015194 IC50 = 650 nM T25315 CA87ZB 90015254 IC50 = 1350 nM T25315 CAK7Q1 90066098 IC50 = 54 nM T25315 CF5L9K 90066144 IC50 = 91 nM T25315 C6ENV5 100951623 EC50 > 10000 nM T25315 C5S3FA 121292609 IC50 = 58 nM T25315 CV02LK 121292615 IC50 = 97 nM T25315 C9FH4Y 121292620 IC50 = 78 nM T25315 C1PK5J 121292622 IC50 = 32 nM T25315 CNM0Z1 121292625 IC50 = 19 nM T25315 CJV62Q 122471809 IC50 = 52 nM T25315 C1X6AT 127030692 EC50 = 600 nM T25315 CRHW82 127030693 EC50 = 758.58 nM T25315 C0J8LG 127030984 EC50 = 194.98 nM T25315 C4G6LB 127030985 EC50 = 229.09 nM T25315 CBA4V3 127030990 EC50 = 165.96 nM T25315 CVX0W5 127030991 EC50 = 512.86 nM T25315 C6JZY5 127031312 EC50 = 6025.6 nM T25315 C6WLS8 127031313 EC50 = 1230.27 nM T25315 C06IOQ 127031899 EC50 = 112.2 nM T25315 CC64XZ 127031900 EC50 = 9.772 nM T25315 C93HLB 127032163 EC50 = 158.49 nM T25315 CKE67A 127032165 EC50 = 125.89 nM T25315 CN38ZL 127032168 EC50 = 158.49 nM T25315 CKV42D 127032453 EC50 = 50.12 nM T25315 C1XSW6 127032454 EC50 = 8511.38 nM T25315 CMO31X 127032455 EC50 = 61.66 nM T25315 C0BZ6S 127032486 EC50 = 58.88 nM T25315 CL8Q5K 127032747 EC50 = 1318.26 nM T25315 CS1JN2 127032750 EC50 = 144.54 nM T25315 CUMG10 134131691 IC50 = 38 nM T25315 CEV3H8 134131840 IC50 = 202 nM T25315 CPC09W 134132003 IC50 = 1300 nM T25315 CKR13E 134132613 IC50 = 70 nM T25315 CQ2C9B 134132726 IC50 = 6600 nM T25315 CU78OH 134134300 IC50 = 340 nM T25315 CO71EK 134134604 IC50 = 4200 nM T25315 CNJ36D 134134840 IC50 = 290 nM T25315 CB9T4J 134134906 IC50 = 40 nM T25315 CC08FB 134135177 IC50 = 330 nM T25315 CAZ6K3 134136033 IC50 = 130 nM T25315 C1SA5H 134136200 IC50 = 225 nM T25315 CPQ65D 134137191 IC50 = 154 nM T25315 CNV52M 134137815 IC50 = 840 nM T25315 CZ4LV2 134137862 IC50 = 2200 nM T25315 CZC36F 134137981 IC50 = 190 nM T25315 C1GP4F 134138894 IC50 = 97 nM T25315 C46FKA 134139917 IC50 = 202 nM T25315 CND4Z9 134140161 IC50 = 82 nM T25315 C1L8KV 134140355 IC50 = 77 nM T25315 CQU74A 134140422 IC50 = 60 nM T25315 CD8HT5 134140497 IC50 = 110 nM T25315 CCPM57 134140635 IC50 = 138 nM T25315 CF41GA 134142277 IC50 = 36 nM T25315 C4DSH2 134143368 IC50 = 403 nM T25315 C9NW5Z 134145083 IC50 = 345 nM T25315 CKJ7I5 134145500 IC50 = 160 nM T25315 C2TYL4 134146441 IC50 = 121 nM T25315 CWJA75 134146842 IC50 = 120 nM T25315 C8RNK1 134147361 IC50 = 790 nM T25315 CJ0BG7 134147406 IC50 = 443 nM T25315 C7EUC1 134147547 IC50 = 3260 nM T25315 CWO0M7 134148525 IC50 = 1200 nM T25315 C6H7FC 134149982 IC50 = 110 nM T25315 CBJ4F7 134150725 IC50 = 1800 nM T25315 CCN4V5 134150746 IC50 = 187 nM T25315 CL7X9S 134150776 IC50 = 780 nM T25315 C68HZQ 134151426 IC50 = 230 nM T25315 CGMB02 134151603 IC50 = 382 nM T25315 C4CA8F 134153150 IC50 = 120 nM T25315 CBL28D 134153156 IC50 = 55 nM T25315 C2RI7V 134153689 IC50 = 65 nM T25315 CX5HE7 134155138 IC50 = 240 nM T25315 COE60H 134156130 IC50 = 105 nM T25315 CHG9K2 134156221 IC50 = 210 nM T25315 C3UM0P 134156632 IC50 = 126 nM T25315 C4C1BX 134157695 IC50 = 39 nM T25315 C6HAX2 136037880 IC50 = 760 nM T25315 D05EML 21847 IC50 > 10000 nM T25315 D0A8PV 45784923 IC50 = 5 nM T25315 D0EK9K 11997335 IC50 = 2.8 nM T89988 D0L5RW 65015 IC50 = 0.04 nM T89988 D00XBC 46861584 IC50 > 10000 nM T89988 D01UBY 46208367 IC50 = 30 nM T89988 D03KKR 3547 IC50 = 35000 nM T89988 D06EPO 11192346 IC50 = 0.5 nM T89988 D06IME 25134303 IC50 = 5 nM T89988 D0O2XQ 11256587 IC50 > 10000 nM T89988 D0TG9Q 11180808 Ki = 0.55 nM T89988 D0YQ7U 11285792 IC50 = 5.9 nM T89988 D0X4SI 9953769 Ki = 58.88 nM T89988 D07KIJ 10008367 IC50 = 3.8 nM T89988 D0Q2JS 10436045 Ki = 16.6 nM T89988 D0W0LS 183789 IC50 = 0.08 nM T89988 C9KT7Q 163751 IC50 = 35000 nM T89988 CJ8NY6 261407 IC50 = 1700 nM T89988 CQ3KO7 483339 IC50 > 1000 nM T89988 C7AP9W 483340 IC50 > 1000 nM T89988 CAB79M 483341 IC50 > 1000 nM T89988 C7XW2D 483342 IC50 > 1000 nM T89988 C7PMT6 483343 IC50 > 1000 nM T89988 CP25RI 483344 IC50 > 1000 nM T89988 CA5BZ8 491773 IC50 > 10000 nM T89988 C0KB6Y 508727 IC50 = 4330 nM T89988 C9J5OC 508729 IC50 = 832 nM T89988 CI96OK 508741 IC50 = 3170 nM T89988 C5P1IN 508742 IC50 = 121 nM T89988 C6B5MG 508744 IC50 = 66000 nM T89988 CRN41P 508749 IC50 = 5500 nM T89988 CEF6L0 508750 EC50 = 40 nM T89988 CUJ2K6 508869 IC50 = 3.9 nM T89988 CAZC09 508870 IC50 = 96 nM T89988 CT83OL 508877 IC50 = 39 nM T89988 CUK86N 3013430 Ki = 23.99 nM T89988 C1TX2Y 3794409 Ki = 199.53 nM T89988 CPZ6S1 3796276 Ki = 213.8 nM T89988 CMT8K7 5481702 IC50 = 10000 nM T89988 CHCY06 6918496 IC50 > 1000 nM T89988 C02HZB 9825735 IC50 = 1500 nM T89988 C9C8EY 9836178 IC50 = 30000 nM T89988 CHP4O1 9840006 IC50 = 1000 nM T89988 CBVJ87 9842404 IC50 = 42000 nM T89988 CH57DZ 9850318 IC50 = 2 nM T89988 C0RB2U 9851741 IC50 = 59 nM T89988 CV58QE 9852285 IC50 = 460 nM T89988 C5XMP4 9857714 IC50 = 2000 nM T89988 CC9U3T 9857981 Ki = 79.43 nM T89988 C56GPV 9858433 IC50 = 4000 nM T89988 C4JEY6 9870980 Ki = 125.89 nM T89988 C9FO1Q 9873546 IC50 = 150 nM T89988 C0PW6L 9885442 IC50 = 390 nM T89988 CZ1OG4 9885683 IC50 = 1020 nM T89988 C8LX2W 9889422 IC50 = 370 nM T89988 C1Q2IG 9890559 IC50 = 13000 nM T89988 C0T6NW 9900683 IC50 = 10000 nM T89988 CC1J0A 9900997 IC50 > 100000 nM T89988 C2R6KA 9902204 Ki = 18.62 nM T89988 C0RH2D 9902578 Ki = 138.04 nM T89988 C9Q6NK 9923015 IC50 = 1600 nM T89988 CY4B8U 9924108 Ki = 162.18 nM T89988 C3Y0QF 9924357 IC50 > 10000 nM T89988 CWG28E 9934977 IC50 = 200 nM T89988 CSH40U 9936494 IC50 > 10000 nM T89988 C7LY1M 9945265 Ki = 95.5 nM T89988 C2KXZ6 9945514 IC50 > 10000 nM T89988 C3PU5K 9946967 IC50 > 10000 nM T89988 CM28YJ 9949615 Ki = 29 nM T89988 CR1Z2G 9952114 IC50 = 6900 nM T89988 C91RTG 9956238 IC50 = 80 nM T89988 C0MGT8 9956260 IC50 = 970 nM T89988 CL3KT8 9967166 Ki = 64.57 nM T89988 CTFZ89 9967349 Ki = 36.31 nM T89988 CBVP31 9967465 Ki = 239 nM T89988 CY89AV 9967878 IC50 = 1000 nM T89988 CA74YF 9974356 IC50 = 11000 nM T89988 CT1FH0 9986630 IC50 = 2.3 nM T89988 CE7IB5 10007642 IC50 = 2.3 nM T89988 C9POK8 10025168 IC50 = 7400 nM T89988 CI3Q9B 10030247 IC50 = 44 nM T89988 C1X6HO 10041590 IC50 = 14000 nM T89988 C5GPK2 10052388 IC50 = 7.798 nM T89988 CQ7N3R 10064487 IC50 = 15000 nM T89988 CMSQ48 10065796 IC50 = 10000 nM T89988 CC03WA 10111333 Ki = 5.623 nM T89988 CM4P8A 10115566 IC50 = 540 nM T89988 C49DEF 10117347 IC50 > 30000 nM T89988 CIDS73 10117480 IC50 = 32 nM T89988 C2ICH4 10119551 IC50 = 28 nM T89988 CC5H0K 10120067 IC50 = 33 nM T89988 C7I9OB 10120907 IC50 = 2.1 nM T89988 CHFP31 10129107 IC50 = 153 nM T89988 CY4AK3 10129192 IC50 = 0.7 nM T89988 CU96TE 10129343 IC50 = 6.5 nM T89988 CM48CP 10132885 Ki = 154.88 nM T89988 CFH9U0 10133557 Ki = 91.2 nM T89988 CF25OU 10137967 IC50 = 320 nM T89988 C47VWF 10138789 IC50 = 630 nM T89988 CAP8K0 10139782 IC50 = 390 nM T89988 CO65TA 10141379 IC50 = 350 nM T89988 C4SHX2 10142792 IC50 = 8 nM T89988 CH83KL 10143025 IC50 = 1200 nM T89988 C09XVI 10144709 IC50 = 1.3 nM T89988 CP6NQ5 10152864 IC50 = 7.5 nM T89988 CF2ZP9 10153373 IC50 = 199.5 nM T89988 CK0CY4 10153431 IC50 = 46 nM T89988 C0Q5AE 10154434 IC50 = 1000 nM T89988 CXI9T2 10154979 IC50 = 1500 nM T89988 C2U4WP 10159217 IC50 > 30000 nM T89988 C93BOF 10161975 IC50 = 1000 nM T89988 CLS30W 10162782 IC50 = 240 nM T89988 CFLN89 10162844 IC50 = 17 nM T89988 CY4OA2 10164316 IC50 = 48 nM T89988 CFKN38 10164641 IC50 > 1000 nM T89988 C50XKS 10165042 IC50 = 190 nM T89988 CKAH17 10165625 IC50 = 5.3 nM T89988 C4V5KG 10165716 IC50 = 150 nM T89988 COMN76 10167417 IC50 = 5.2 nM T89988 CI45NC 10175423 IC50 = 21 nM T89988 C10HSL 10175425 IC50 = 1.4 nM T89988 CBTG57 10182382 IC50 = 66 nM T89988 C1BGH8 10182763 IC50 > 30000 nM T89988 CH5AC1 10183362 IC50 = 64 nM T89988 CGP07U 10184007 IC50 = 1190 nM T89988 C2ED3X 10184169 IC50 > 10000 nM T89988 C5A2QV 10184250 IC50 = 100 nM T89988 CM80RH 10186010 IC50 = 100 nM T89988 C5Z8RT 10187492 IC50 = 84 nM T89988 C89VMQ 10195882 IC50 = 37 nM T89988 CSM35L 10196988 IC50 = 38 nM T89988 C9SX8I 10203447 IC50 = 2200 nM T89988 CXK43P 10204589 IC50 > 30000 nM T89988 C4OM2Z 10205915 IC50 > 10000 nM T89988 CNI37B 10205937 IC50 = 110 nM T89988 CWZY76 10206007 IC50 = 65 nM T89988 CV5WX9 10206776 IC50 = 170 nM T89988 CS0RU7 10207542 IC50 = 87 nM T89988 CM0UY9 10207590 IC50 = 19 nM T89988 CH04CE 10207591 IC50 = 600 nM T89988 CS98YN 10207639 IC50 = 11 nM T89988 CWC7X1 10208080 IC50 > 10000 nM T89988 CHDE08 10208555 IC50 = 6400 nM T89988 C4NMH6 10208946 IC50 = 27 nM T89988 C6YL0V 10209102 IC50 = 7000 nM T89988 C91ZMU 10209478 IC50 = 5 nM T89988 CE4I6T 10218403 IC50 = 1.5 nM T89988 CO48MN 10218812 IC50 = 41.3 nM T89988 CHP92E 10218843 IC50 = 8.4 nM T89988 C4EBQ9 10225909 IC50 = 5500 nM T89988 CF3WZ0 10227556 IC50 = 250 nM T89988 C84HKV 10227655 IC50 = 160 nM T89988 CK9AQ7 10228205 IC50 = 88 nM T89988 CYV95X 10228435 IC50 = 7 nM T89988 C72HMR 10228761 IC50 > 30000 nM T89988 C02UNG 10232019 IC50 = 9.3 nM T89988 CV7G6W 10239671 IC50 = 172 nM T89988 CMF6D0 10239991 IC50 = 2.05 nM T89988 C1AK9C 10240064 IC50 = 0.2 nM T89988 CU53XR 10240278 IC50 = 44.5 nM T89988 C3H4ST 10245340 IC50 = 30000 nM T89988 CNEW23 10256127 IC50 = 1230 nM T89988 CMRA02 10257042 Ki = 39.81 nM T89988 CPX15I 10268598 IC50 = 3900 nM T89988 CR6SA7 10269886 IC50 > 10000 nM T89988 CK49NQ 10272003 IC50 = 700 nM T89988 CPOD91 10276594 IC50 = 230 nM T89988 CIHB65 10277182 IC50 = 3010 nM T89988 C3CZ7H 10277466 IC50 > 10000 nM T89988 CO2HE6 10278257 IC50 = 19 nM T89988 CWGJ31 10278862 IC50 = 97 nM T89988 CW0H9D 10279078 IC50 = 41 nM T89988 CXZ08C 10279914 IC50 = 2400 nM T89988 CE9ID0 10280944 IC50 > 10000 nM T89988 CD4YG9 10281316 IC50 = 3.6 nM T89988 CWGK21 10281715 IC50 = 4.7 nM T89988 C7ODM2 10289827 IC50 = 0.3 nM T89988 CH97RC 10291634 IC50 = 1500 nM T89988 CDU26C 10293022 Ki = 15.85 nM T89988 CJ06NI 10299408 IC50 = 31 nM T89988 C6E1CB 10299952 IC50 = 400 nM T89988 C06FDK 10300282 IC50 = 110 nM T89988 CFX3M7 10300284 IC50 = 6.7 nM T89988 C6LP8U 10300705 IC50 = 7860 nM T89988 CO0P4F 10301330 IC50 > 10000 nM T89988 CDRW29 10302973 IC50 = 65 nM T89988 CF01AR 10304021 IC50 = 4 nM T89988 CY7P9S 10312346 IC50 = 8.1 nM T89988 C2QM0N 10315045 IC50 = 17000 nM T89988 CWFB30 10323427 IC50 = 30 nM T89988 CCDY38 10323468 IC50 = 28 nM T89988 CBA2C6 10325032 IC50 = 6 nM T89988 C1N0CE 10346048 IC50 = 173.78 nM T89988 CT40XZ 10348168 IC50 = 165 nM T89988 C62PXQ 10360623 IC50 = 23000 nM T89988 CC0YO3 10371682 IC50 = 1040 nM T89988 C7PUE4 10392559 IC50 = 64 nM T89988 CCZ17H 10392978 IC50 = 2 nM T89988 CU81IS 10409097 IC50 = 30000 nM T89988 CKYF72 10414966 IC50 = 144 nM T89988 CZ65IG 10427217 IC50 = 14000 nM T89988 C6GQ5E 10427222 IC50 = 56 nM T89988 CYVI63 10436083 IC50 = 400 nM T89988 C8SPW7 10458152 IC50 = 218.78 nM T89988 CI10WZ 10459336 IC50 = 900 nM T89988 C9NZT2 10471319 IC50 = 22000 nM T89988 CJL0P6 10482463 IC50 = 50 nM T89988 C95LRC 10940216 Ki = 590 nM T89988 CQ6S7M 10957890 IC50 = 2000 nM T89988 CR52KG 11155781 IC50 = 49 nM T89988 C8BF7M 11179439 IC50 = 3.8 nM T89988 CAEB68 11180383 IC50 = 7.9 nM T89988 CZ80GK 11180885 IC50 = 240 nM T89988 C1KHV0 11192300 IC50 = 40 nM T89988 C16MCS 11192943 IC50 = 0.9 nM T89988 CG9OA2 11214277 IC50 = 305 nM T89988 CTN5C2 11215504 IC50 = 340 nM T89988 CK21LX 11223594 IC50 > 10000 nM T89988 C62UXT 11226430 IC50 = 20 nM T89988 CU75LJ 11227168 IC50 = 4.3 nM T89988 C5AYG7 11227368 IC50 = 102 nM T89988 CO3M2S 11227383 IC50 = 125 nM T89988 CA39QR 11227406 IC50 > 10000 nM T89988 C3G5PZ 11237168 IC50 = 65 nM T89988 C1LWU2 11237256 IC50 = 43 nM T89988 CQ6KW0 11272103 IC50 = 10000 nM T89988 CZ8DU0 11273379 IC50 = 8.8 nM T89988 CTRB13 11273475 IC50 = 131.5 nM T89988 CSG19P 11283842 IC50 = 4.5 nM T89988 C06TUD 11285791 IC50 = 5.9 nM T89988 C7N1ZH 11296325 IC50 = 53 nM T89988 C0P9IM 11296618 IC50 = 51.5 nM T89988 CA63BF 11306757 IC50 = 7.1 nM T89988 CW47VZ 11318368 IC50 = 95 nM T89988 C4FS8T 11319072 IC50 = 10 nM T89988 C1A5ET 11329244 IC50 = 10000 nM T89988 CGE2P7 11329328 IC50 = 126 nM T89988 CQ1CG9 11330529 IC50 = 5.4 nM T89988 CIT2Y7 11330837 IC50 = 10 nM T89988 CX3PY4 11340816 IC50 = 66 nM T89988 C95SAU 11341950 IC50 = 710 nM T89988 CF98IO 11342351 IC50 = 38 nM T89988 CKZ20A 11353843 IC50 = 3.6 nM T89988 CX6C2M 11353855 IC50 = 1.9 nM T89988 C0JT3P 11364218 IC50 = 217 nM T89988 CZ82WH 11365166 IC50 = 1.8 nM T89988 CE2M9F 11387511 IC50 = 2.6 nM T89988 CE5ZK6 11409228 IC50 = 11 nM T89988 C2N0AG 11421712 IC50 = 3.8 nM T89988 CWV9L6 11421840 IC50 = 2.8 nM T89988 C9Z0TH 11433008 IC50 = 2.4 nM T89988 C1K6PE 11456448 IC50 = 45.5 nM T89988 CH7E4M 11466237 IC50 = 51 nM T89988 C25XGJ 11467577 IC50 = 136.5 nM T89988 C3S7DQ 11478362 IC50 = 690 nM T89988 C78GWT 11489078 IC50 = 23 nM T89988 C70LYJ 11497533 IC50 = 15 nM T89988 C7I8FQ 11502188 IC50 = 1184 nM T89988 C40IMW 11502371 IC50 = 20 nM T89988 CB7UX1 11504634 IC50 = 17 nM T89988 C1LCD7 11510932 IC50 = 244 nM T89988 CWVX78 11512375 IC50 = 16.7 nM T89988 C54PDI 11526729 IC50 = 50 nM T89988 C0BF5R 11527661 IC50 = 2.6 nM T89988 C0F7SR 11534473 IC50 = 6 nM T89988 CG29EI 11540494 IC50 = 0.6 nM T89988 C4AH1P 11541149 IC50 = 15 nM T89988 C0HYO4 11548199 IC50 = 2 nM T89988 CKGI84 11553070 IC50 = 37 nM T89988 C26UCI 11553489 IC50 = 15 nM T89988 CK5DE0 11555541 IC50 = 40 nM T89988 CCJ4G1 11555827 IC50 = 2.5 nM T89988 C9HK2R 11562947 IC50 = 10 nM T89988 C4E7NT 11563451 IC50 = 178 nM T89988 C5AL9R 11563597 IC50 = 633.87 nM T89988 CCQ8O9 11567495 IC50 = 123 nM T89988 CQ0TD1 11570045 IC50 = 441.57 nM T89988 CLY5O2 11570431 IC50 = 209 nM T89988 C7RKT1 11577400 IC50 = 213 nM T89988 C2DG4A 11582651 IC50 = 161 nM T89988 C41DRT 11584094 IC50 = 6 nM T89988 C6KL3Q 11585168 IC50 = 43.95 nM T89988 CBN18P 11590644 IC50 = 567 nM T89988 CYG74X 11591595 IC50 = 7 nM T89988 CF50KQ 11591776 IC50 = 5 nM T89988 CN5OV9 11591956 IC50 = 4 nM T89988 CH0OD8 11598084 IC50 = 42 nM T89988 C1DKF4 11598797 IC50 > 10000 nM T89988 C1FH6B 11599317 IC50 = 7 nM T89988 C9FK3O 11605635 IC50 = 6 nM T89988 C6BET5 11605867 IC50 = 20 nM T89988 CYP0L5 11605985 IC50 = 522.4 nM T89988 CS8HR5 11606147 IC50 = 10 nM T89988 CZQ78X 11606167 IC50 = 2391 nM T89988 C84YPR 11606411 IC50 = 1.3 nM T89988 C6V9WA 11606702 IC50 = 8.995 nM T89988 CTQ6D9 11613399 IC50 = 6 nM T89988 C1N4CJ 11620726 IC50 = 167.88 nM T89988 CS9R1X 11621035 IC50 = 7.7 nM T89988 C8NKD4 11627639 IC50 = 2.4 nM T89988 C05TNG 11627840 IC50 = 0.2 nM T89988 CNS5P7 11632418 IC50 = 170 nM T89988 C40GEC 11633080 IC50 = 90 nM T89988 CU7B6I 11634118 IC50 = 904 nM T89988 C3EAG5 11634928 IC50 = 9 nM T89988 C57RHQ 11634966 IC50 > 10000 nM T89988 C2OD0U 11635092 IC50 = 120 nM T89988 CQ65EJ 11640044 IC50 = 30 nM T89988 CP21CA 11641253 IC50 = 46 nM T89988 C0B9YV 11643006 IC50 = 0.6 nM T89988 C9IOM8 11647276 IC50 = 16 nM T89988 C3IFQ9 11662833 IC50 = 80 nM T89988 CU7RT2 11663882 IC50 = 10 nM T89988 CNJE21 11663995 IC50 = 1225 nM T89988 CU7OG2 11669935 IC50 = 18 nM T89988 CPI1S3 11670910 IC50 = 1800 nM T89988 CC2LB1 11670968 IC50 = 25 nM T89988 CVX87R 11671120 IC50 = 50 nM T89988 C6BY1A 11678573 IC50 = 66 nM T89988 CR91QA 11690139 IC50 = 856 nM T89988 CS1W5I 11690536 IC50 = 337 nM T89988 CJL2T5 11692057 IC50 = 210 nM T89988 CS31YE 11699149 IC50 = 4 nM T89988 C4QLY1 11699524 IC50 = 6 nM T89988 CI5G6C 11699541 IC50 = 20 nM T89988 CU8L6Q 11700079 IC50 = 6.3 nM T89988 CCB51S 11706775 IC50 = 207.01 nM T89988 C6CM7S 11711078 IC50 = 277 nM T89988 CJ03AX 11712754 IC50 = 40 nM T89988 C9IQK5 11713221 IC50 = 10 nM T89988 CDN6X8 11718088 IC50 = 40 nM T89988 CKF6U5 11721085 IC50 = 30 nM T89988 C38IBK 11721374 IC50 = 1 nM T89988 CZR39O 11723420 IC50 = 20000 nM T89988 CPG15O 11743399 IC50 > 10000 nM T89988 C4L9EC 11752457 IC50 = 6.9 nM T89988 C7A4YV 11753466 IC50 = 1.9 nM T89988 CU5P8D 11753664 IC50 = 11 nM T89988 CKW9D4 11756884 IC50 = 2.3 nM T89988 C1S3JD 11843812 IC50 = 822 nM T89988 C2X7GJ 11843813 IC50 = 930 nM T89988 CS6JC4 11843945 IC50 = 1000 nM T89988 CBV2X9 11843946 IC50 = 1100 nM T89988 C1HV9G 11844079 IC50 = 1100 nM T89988 CR7MI5 11844083 IC50 = 780 nM T89988 CEM02F 11844209 IC50 = 160 nM T89988 C2J8RH 11844212 IC50 = 80 nM T89988 C02CKY 11844329 IC50 = 320 nM T89988 C9RE0B 11844467 IC50 = 1500 nM T89988 C63QMF 11844468 IC50 = 700 nM T89988 C0DRU3 11844469 IC50 = 140 nM T89988 CGHL19 11844470 IC50 = 45 nM T89988 C5PL9R 11844471 IC50 = 440 nM T89988 CMT8N9 11844595 IC50 = 120 nM T89988 CRY83B 12093162 Ki = 213.8 nM T89988 C2QWR3 12093163 Ki = 263.03 nM T89988 C79CBJ 12093167 Ki = 10 nM T89988 CJX31Q 12093170 IC50 = 170 nM T89988 CH5QK9 15290299 IC50 = 230 nM T89988 C1T0SU 15518124 IC50 = 13400 nM T89988 C7X3CQ 15604497 Ki = 25.12 nM T89988 CQJ7Y2 15985912 Ki = 10 nM T89988 C0G1SC 15985914 Ki = 31.62 nM T89988 CKE0U5 15985981 Ki = 501.19 nM T89988 CYA3K5 16064151 IC50 = 0.4 nM T89988 CX04NO 16066354 IC50 = 1.7 nM T89988 C9G8TZ 16124598 Ki = 1.259 nM T89988 CH90BN 16216716 IC50 = 1.8 nM T89988 C6D5FS 16720313 IC50 = 36 nM T89988 C9XH8N 17756652 Ki = 10 nM T89988 CMEZ85 17838131 IC50 > 100000 nM T89988 CGFW16 17838175 IC50 > 100000 nM T89988 CZT35Q 17838190 IC50 > 100000 nM T89988 CCR8J4 17838276 IC50 > 100000 nM T89988 C5CH8K 17866152 IC50 = 5000 nM T89988 CMD76W 18426157 IC50 = 17000 nM T89988 C0EB8U 18426192 IC50 = 11000 nM T89988 CRM90U 19430534 Ki = 794.33 nM T89988 C6K9RC 21098468 IC50 = 8000 nM T89988 CMF27K 21098469 IC50 = 7000 nM T89988 C7WBX4 21098475 IC50 > 30000 nM T89988 CFB3T6 21098478 IC50 = 8000 nM T89988 C9T8FA 21098480 IC50 = 5000 nM T89988 CMA42E 21098488 IC50 = 1000 nM T89988 C9JI3T 21098490 IC50 = 1000 nM T89988 CK51MC 21098512 IC50 = 19000 nM T89988 CN8F1W 21098519 IC50 = 1000 nM T89988 CW0BP6 21098523 IC50 = 1000 nM T89988 C1WM8S 21098530 IC50 = 19000 nM T89988 CYX26M 22143104 IC50 = 19 nM T89988 CF9I5G 22143112 IC50 = 3.8 nM T89988 C10IVJ 22143146 IC50 = 5.5 nM T89988 C8ESY2 22143155 IC50 = 5.4 nM T89988 C53NIP 22143196 IC50 = 28 nM T89988 C5G7CR 22143200 IC50 = 510 nM T89988 CZ3BU6 22143225 IC50 = 167.5 nM T89988 C17DEU 22143241 IC50 = 7 nM T89988 CDB86Q 22143255 IC50 = 2 nM T89988 C8LDZ2 22143258 IC50 = 22.5 nM T89988 CX1L8K 22143293 IC50 = 6.1 nM T89988 CH85XV 22143294 IC50 = 7.9 nM T89988 C89IFO 22143305 IC50 = 12.5 nM T89988 CY4GU1 22143308 IC50 = 123 nM T89988 CVZ64R 22143309 IC50 = 26 nM T89988 CV8F9U 22143314 IC50 = 463 nM T89988 C42ZHE 22143334 IC50 = 0.95 nM T89988 CP6X1V 22143346 IC50 = 4.8 nM T89988 C3POB6 22143349 IC50 = 155 nM T89988 C2CPY8 22268768 IC50 = 8700 nM T89988 C1TS9Z 22310839 IC50 = 2200 nM T89988 CT36VS 22310850 IC50 = 8600 nM T89988 CT4C1M 22310869 IC50 = 2300 nM T89988 CRX1D6 22310876 IC50 = 6090 nM T89988 CM2S9I 22310877 IC50 = 1130 nM T89988 C7ZJ3B 22310883 IC50 = 230 nM T89988 CI1C9R 22310896 IC50 = 170 nM T89988 C7GH1P 22310899 IC50 = 1360 nM T89988 C59BIA 22310903 IC50 = 1210 nM T89988 CG25OW 22310914 IC50 = 90 nM T89988 CDY16V 22310924 IC50 = 340 nM T89988 CG8L6I 22310929 IC50 = 125 nM T89988 C9E4LG 22310939 IC50 = 1050 nM T89988 C6R0DG 22310943 IC50 = 1640 nM T89988 CKY2B0 22310945 IC50 = 410 nM T89988 CFQ7P1 22310946 IC50 = 1310 nM T89988 C64QRB 22310953 IC50 = 1270 nM T89988 C3P8YN 22310954 IC50 = 110 nM T89988 C6D4KC 22310965 IC50 = 99 nM T89988 CW37TA 22310971 IC50 = 1190 nM T89988 C0CZL1 22310972 IC50 = 640 nM T89988 CUG43R 22310976 IC50 = 150 nM T89988 C38PHN 22310991 IC50 = 280 nM T89988 CJ2H7Q 22310992 IC50 = 96 nM T89988 C8RPO2 22310995 IC50 = 500 nM T89988 CE32SQ 22311000 IC50 = 340 nM T89988 CTV2K4 22311005 IC50 = 4780 nM T89988 CC9YA1 22335665 Ki = 57 nM T89988 CTO2A8 22335694 Ki = 17.78 nM T89988 C2NK9E 22394337 IC50 = 3010 nM T89988 CKO01W 22725647 Ki = 8.128 nM T89988 CT7Q3X 23405932 IC50 = 55 nM T89988 CB28YR 23441036 IC50 = 21000 nM T89988 CZA0F3 23441058 IC50 = 19000 nM T89988 CUI9H4 23630215 IC50 = 7.3 nM T89988 CEP68R 23655673 IC50 = 3300 nM T89988 C4BZ9J 23655877 IC50 = 1100 nM T89988 C6BDU5 23656067 IC50 = 470 nM T89988 C53TJN 23656260 IC50 = 660 nM T89988 CL0GR2 23656261 IC50 = 115 nM T89988 CZ05MF 23656430 IC50 = 4 nM T89988 C2LOI1 23656431 IC50 = 4 nM T89988 C5JNY2 23656432 IC50 = 3400 nM T89988 C0WBE1 23656433 IC50 = 6800 nM T89988 C98MGF 23656434 IC50 = 720 nM T89988 CM5SO9 23656584 IC50 = 320 nM T89988 CN9GW5 23656585 IC50 = 210 nM T89988 C7JV4W 23725177 IC50 = 0.67 nM T89988 C25HKJ 24758044 IC50 > 20000 nM T89988 C4QO9W 24801178 IC50 = 12000 nM T89988 C9P3YJ 24801179 IC50 = 2170 nM T89988 CT05NH 24801180 IC50 = 2117.2 nM T89988 C8Q4KT 24801342 IC50 = 530 nM T89988 CV28RW 24801343 IC50 = 400 nM T89988 C9NT2S 24801344 IC50 = 360 nM T89988 C5RV7A 24801345 IC50 = 4130 nM T89988 CI1EC7 24801346 IC50 = 550 nM T89988 CM81GS 24801522 IC50 = 37 nM T89988 CXYQ23 24801523 IC50 = 64 nM T89988 C64WPY 24801524 IC50 = 87 nM T89988 C9EB2J 24801525 IC50 = 130 nM T89988 C4C2LP 24801526 IC50 = 4.8 nM T89988 CKW46B 24801689 IC50 = 9 nM T89988 CA15KP 24801690 IC50 = 5.1 nM T89988 C3K1DA 25007995 IC50 = 80 nM T89988 CB45YS 25007996 IC50 = 160 nM T89988 CM17BE 25008678 IC50 = 6450 nM T89988 CU69WN 25008679 IC50 = 12000 nM T89988 C4OH9R 25008849 IC50 = 8400 nM T89988 C0HIK4 25010616 IC50 = 160 nM T89988 C9W6LE 25022597 IC50 = 3.2 nM T89988 CDKJ78 25033361 IC50 = 300 nM T89988 CLM02V 25110564 Ki = 5300 nM T89988 CGO4J0 25110660 Ki = 79 nM T89988 C9XI0Q 25110678 Ki = 7100 nM T89988 CKA50N 25110679 Ki = 5100 nM T89988 C3SHW4 25110716 IC50 = 2.5 nM T89988 C6U3YK 25110788 IC50 = 3 nM T89988 C67QXP 25154827 IC50 = 4 nM T89988 C54LQF 25230828 IC50 > 50000 nM T89988 CK5HZ8 25256791 IC50 = 1200 nM T89988 C8IHN4 25267730 IC50 = 1020 nM T89988 C50IVN 25267738 IC50 = 4750 nM T89988 C0ZVT1 25268077 IC50 > 10000 nM T89988 CJD3B9 25268081 IC50 = 200 nM T89988 CR9M5T 25268085 IC50 = 250 nM T89988 CZ3BX9 25268434 IC50 > 10000 nM T89988 CT5XC3 25268436 IC50 = 390 nM T89988 CKA42N 25268440 IC50 = 230 nM T89988 CC3Y9N 25268442 IC50 = 9550 nM T89988 C0O3DW 25268795 IC50 = 8950 nM T89988 CK03BL 25268803 IC50 = 1810 nM T89988 C41GLE 25269516 IC50 = 4250 nM T89988 CLZ9P0 25270182 IC50 = 3440 nM T89988 C2FZ9P 42606792 IC50 = 1.8 nM T89988 C1VQ0H 42632811 IC50 = 11350 nM T89988 C2L3AW 42632830 IC50 = 7800 nM T89988 COGL90 42632836 IC50 = 710 nM T89988 CTDE24 42632840 IC50 = 3250 nM T89988 CYLQ82 42632863 IC50 = 2000 nM T89988 CB95UT 42632867 IC50 > 10000 nM T89988 CLCX87 42632888 IC50 = 2550 nM T89988 CU2PO5 44180522 Ki = 6 nM T89988 C5YFB9 44252324 IC50 > 10000 nM T89988 C13YRA 44296077 Ki = 5900 nM T89988 CTN90Y 44296087 Ki = 420 nM T89988 CTNF31 44296137 Ki = 79 nM T89988 CR1WU3 44296138 Ki > 10000 nM T89988 C9D4HM 44296154 Ki = 660 nM T89988 CKU4Y6 44296155 Ki = 2500 nM T89988 CSTN01 44296156 Ki > 10000 nM T89988 CD53WG 44296219 IC50 = 32 nM T89988 CL5VC0 44296240 Ki > 10000 nM T89988 CJGP84 44296264 Ki = 1700 nM T89988 C0IT6Z 44296265 Ki = 1450 nM T89988 CUG58H 44296266 Ki = 790 nM T89988 C1ZT7N 44296268 Ki = 234 nM T89988 C4M5CB 44296269 Ki = 2800 nM T89988 CX2U4R 44296287 Ki = 2900 nM T89988 CKD7I3 44296309 Ki = 6300 nM T89988 CVG7F2 44296310 Ki = 1200 nM T89988 CG0YU3 44296344 Ki = 4200 nM T89988 C52TFI 44296366 Ki = 360 nM T89988 C9VQ3K 44296384 Ki = 360 nM T89988 CAK80S 44296398 Ki = 550 nM T89988 CW5M1B 44296409 Ki = 4400 nM T89988 C02RMO 44296410 Ki = 560 nM T89988 CUY1A6 44296428 Ki = 520 nM T89988 C1FOD9 44296429 Ki = 870 nM T89988 C4H7XD 44296469 Ki = 4400 nM T89988 CL47OS 44296501 Ki = 1600 nM T89988 C6AR0I 44296628 Ki = 790 nM T89988 CYTQ98 44296629 Ki = 460 nM T89988 C74OLQ 44296630 Ki = 350 nM T89988 C67OGJ 44309012 Ki = 251 nM T89988 CUH16K 44353170 IC50 = 12700 nM T89988 CJ51CI 44353190 IC50 = 770 nM T89988 C4SWE0 44353196 IC50 = 1030 nM T89988 C03UXF 44353197 IC50 = 370 nM T89988 CU4ZX3 44353205 IC50 > 50000 nM T89988 C8X6VI 44353223 IC50 = 27000 nM T89988 CF6SK1 44353334 IC50 = 1480 nM T89988 CQK9U6 44353356 IC50 = 12300 nM T89988 CN7MI9 44353367 IC50 = 300 nM T89988 C2LA3C 44353369 IC50 = 5770 nM T89988 CYMD40 44353370 IC50 = 650 nM T89988 CM1OG0 44353377 IC50 = 3880 nM T89988 C9XGW6 44353380 IC50 > 50000 nM T89988 C4EG3U 44353395 IC50 = 120 nM T89988 CBYQ54 44353396 IC50 = 220 nM T89988 CV54UG 44353408 IC50 > 50000 nM T89988 C5Q3VF 44353418 IC50 = 10840 nM T89988 C2PIM0 44353464 IC50 = 260 nM T89988 CRVF39 44353617 IC50 = 12600 nM T89988 CZE90S 44395028 IC50 = 1500 nM T89988 CYJC04 44395029 IC50 = 2300 nM T89988 CIHC30 44395036 IC50 = 74000 nM T89988 CUFP61 44395048 IC50 = 1500 nM T89988 CGN58X 44395055 EC50 = 610 nM T89988 C1N9IW 44395058 IC50 = 11000 nM T89988 C20DZS 44395061 IC50 = 1500 nM T89988 CJ47HB 44395062 IC50 = 1500 nM T89988 CW78VC 44395066 IC50 = 87000 nM T89988 C2HY0B 44395079 IC50 = 9300 nM T89988 CZ7EM1 44395088 IC50 = 7000 nM T89988 C7HL3J 44395092 IC50 = 6400 nM T89988 CXN1E3 44395093 IC50 = 11000 nM T89988 C1G8LN 44395094 IC50 = 4500 nM T89988 C78EIY 44395097 IC50 = 22000 nM T89988 CC0VD9 44395104 IC50 = 17000 nM T89988 C0EZ1N 44395113 IC50 = 11000 nM T89988 C4P3YI 44395114 IC50 > 100000 nM T89988 CVR3C4 44395125 IC50 = 43000 nM T89988 C17BVS 44395126 IC50 = 710 nM T89988 C98JAY 44395129 IC50 = 40000 nM T89988 CJVK23 44395136 IC50 = 4200 nM T89988 CL9B7U 44395137 IC50 = 34000 nM T89988 C2JKO7 44395138 IC50 = 28000 nM T89988 CI74MR 44395143 IC50 = 41000 nM T89988 C8W7QA 44395144 IC50 = 14000 nM T89988 CQVF83 44395160 IC50 = 19000 nM T89988 C6PO5T 44395165 IC50 = 4000 nM T89988 C0UT4Q 44395169 IC50 = 33000 nM T89988 C58SKQ 44395186 IC50 = 4100 nM T89988 CP4WI3 44395194 IC50 = 12000 nM T89988 CQG0T2 44395195 IC50 = 26000 nM T89988 CC39VA 44395201 IC50 = 64000 nM T89988 CK4RW1 44395222 IC50 = 2400 nM T89988 C2O0XM 44395232 IC50 = 7900 nM T89988 CX81WJ 44395238 IC50 = 7800 nM T89988 C1KR3H 44395239 IC50 = 50000 nM T89988 CBT0O9 44395254 IC50 = 45000 nM T89988 CQC21H 44395256 IC50 = 16000 nM T89988 C72LSP 44413076 IC50 = 8 nM T89988 CG8VJ4 44413089 IC50 = 10 nM T89988 C6R8TI 44413137 IC50 = 865 nM T89988 C2FRX1 44413144 IC50 = 720 nM T89988 C5PA2Q 44413147 IC50 = 424 nM T89988 C03JIF 44413158 IC50 = 592 nM T89988 CXB7S3 44413167 IC50 = 1000 nM T89988 CA35QW 44413214 IC50 = 32 nM T89988 C0LT7X 44413230 IC50 = 1477 nM T89988 CV26LN 44413257 IC50 = 25 nM T89988 C0UL2N 44413258 IC50 = 13 nM T89988 C5J2IA 44413310 IC50 = 678 nM T89988 C39VOA 44413311 IC50 = 521 nM T89988 COD13L 44413328 IC50 = 342 nM T89988 C9EVF0 44413344 IC50 = 575 nM T89988 C07HRT 44413399 IC50 = 831.76 nM T89988 C7W8LI 44413411 IC50 = 756 nM T89988 C71QPH 44414578 IC50 = 1070 nM T89988 CW3V9I 44415864 IC50 = 48 nM T89988 CXQ4E0 44415880 IC50 = 4 nM T89988 CJYB82 44415898 IC50 = 38 nM T89988 CDV84J 44415899 IC50 = 13 nM T89988 C79IPU 44415900 IC50 = 244 nM T89988 CS51WY 44415903 IC50 = 129 nM T89988 CLHX29 44415904 IC50 = 42 nM T89988 CGX2M9 44415922 IC50 = 15 nM T89988 C8KU5F 44415927 IC50 = 216 nM T89988 CVF2X9 44415939 IC50 = 37 nM T89988 C4RCE6 44415942 IC50 = 462 nM T89988 C0FMC7 44415945 IC50 = 437 nM T89988 CYTL74 44415957 IC50 = 86 nM T89988 CYQE71 44415958 IC50 = 73 nM T89988 CKX2L3 44415973 IC50 = 37 nM T89988 CJ51SX 44415992 IC50 = 47 nM T89988 CI38AS 44415995 IC50 = 80 nM T89988 CP4DF0 44415996 IC50 = 298 nM T89988 CF4SD2 44416015 IC50 = 72 nM T89988 COX2Z8 44416041 IC50 = 72 nM T89988 CGKV54 44416066 IC50 = 125 nM T89988 CN8V6W 44416070 IC50 = 525 nM T89988 C5D9UT 44416125 IC50 = 805 nM T89988 C7P5KX 44416138 IC50 = 11 nM T89988 CVTL23 44416156 IC50 = 783 nM T89988 CVMS82 44416157 IC50 = 3 nM T89988 CYR56S 44416273 IC50 = 570 nM T89988 CE7K0V 44416274 IC50 = 213.8 nM T89988 C9OBD5 44421855 IC50 = 20000 nM T89988 CFKZ21 44421856 IC50 > 30000 nM T89988 C7N8YR 44421860 IC50 = 10000 nM T89988 CQW39E 44421862 IC50 = 6000 nM T89988 CQ07XN 44421867 IC50 = 1000 nM T89988 C7SL3R 44421868 IC50 = 5000 nM T89988 C7L2UB 44421888 IC50 = 6000 nM T89988 CUD80R 44421889 IC50 = 1000 nM T89988 C3K7NQ 44421913 IC50 = 1000 nM T89988 C7PCB4 44421917 IC50 = 1000 nM T89988 C5T6WC 44421922 IC50 = 3000 nM T89988 C87DBT 44421923 IC50 = 2000 nM T89988 CZ6DH9 44423281 IC50 = 65 nM T89988 CWJ3C4 44423282 IC50 = 7.5 nM T89988 CKX2F3 44423283 IC50 = 1.4 nM T89988 CJH60R 44423284 IC50 > 1000 nM T89988 CQ80SV 44423285 IC50 = 47 nM T89988 CNR96O 44425241 IC50 = 20 nM T89988 C1DO8P 44425242 IC50 = 9.1 nM T89988 CZ49XH 44425243 IC50 = 28.6 nM T89988 C9POR6 44425244 IC50 = 7.3 nM T89988 CW5B2T 44425245 IC50 = 1.3 nM T89988 CNPT74 44425247 IC50 = 182.7 nM T89988 C9VET7 44425249 IC50 = 5.2 nM T89988 CIK35U 44425250 IC50 = 1.8 nM T89988 C04TAL 44425252 IC50 = 3 nM T89988 CA64XV 44425254 IC50 = 0.7 nM T89988 C0L2CH 44425255 IC50 = 0.6 nM T89988 CK1QL4 44425256 IC50 = 32.7 nM T89988 CJS6E3 44425258 IC50 = 14.5 nM T89988 CHC0X9 44425271 IC50 = 4 nM T89988 CCB89O 44425272 IC50 = 3.5 nM T89988 C46TAL 44425273 IC50 = 3.9 nM T89988 C4N9YV 44425274 IC50 = 7.4 nM T89988 CZWS87 44425276 IC50 = 18 nM T89988 C49VPJ 44425277 IC50 = 16 nM T89988 CR0W5Q 44425279 IC50 = 2.6 nM T89988 CYA4L7 44425281 IC50 = 1.3 nM T89988 C4IE0H 44425283 IC50 = 36 nM T89988 CTH31J 44425286 IC50 = 14.3 nM T89988 CM4D6U 44425288 IC50 = 13.18 nM T89988 CHD4K8 44425290 IC50 = 3.5 nM T89988 C8EXT0 44425292 IC50 = 0.43 nM T89988 CW7E4Z 44425293 IC50 = 1.4 nM T89988 CAF01W 44425294 IC50 = 0.8 nM T89988 C9HNI1 44425304 IC50 = 13.18 nM T89988 CQ7W8I 44425305 IC50 = 229 nM T89988 CPY5O8 44425306 IC50 = 41.69 nM T89988 C59CGR 44425308 IC50 = 30 nM T89988 C7XI6U 44425309 IC50 = 6.5 nM T89988 CG7Z2F 44425310 IC50 = 5.8 nM T89988 C9H1OJ 44425315 IC50 = 13 nM T89988 CT75JS 44425316 IC50 = 17 nM T89988 C4JPK2 44425317 IC50 = 19 nM T89988 CJY1R8 44425318 IC50 = 23 nM T89988 C9DHM6 44425319 IC50 = 13 nM T89988 CG1J9N 44425320 IC50 = 14 nM T89988 CB1IP4 44425321 IC50 = 74 nM T89988 CTQ3W1 44425322 IC50 = 36 nM T89988 C54TVY 44425629 IC50 = 20 nM T89988 CET0P3 44425630 IC50 = 8.913 nM T89988 C2P8SI 44425631 IC50 = 10 nM T89988 CBI1A0 44425633 IC50 = 7.586 nM T89988 CQP64B 44425634 IC50 = 15.85 nM T89988 CQ4H3S 44425635 IC50 = 8 nM T89988 C3KSH7 44425636 IC50 = 20 nM T89988 CJI4T7 44425637 IC50 = 19 nM T89988 CH13ZK 44425638 IC50 = 231 nM T89988 CNY18R 44425639 IC50 = 15.5 nM T89988 C10GTR 44425640 IC50 = 6.5 nM T89988 C6GVI5 44425641 IC50 = 13 nM T89988 CM0SY9 44425642 IC50 = 28 nM T89988 C3T7DE 44425643 IC50 = 3.981 nM T89988 CQL1F7 44425644 IC50 = 3.3 nM T89988 C9PR2I 44425645 IC50 = 0.15 nM T89988 C1IGE8 44425646 IC50 = 5 nM T89988 C3W2SM 44425647 IC50 = 0.32 nM T89988 CXI0Y9 44425648 IC50 = 5.5 nM T89988 CDKA32 44425649 IC50 = 6.3 nM T89988 CQK4M8 44425650 IC50 = 27 nM T89988 CIH7T2 44425651 IC50 = 8.5 nM T89988 C8WXN5 44425652 IC50 = 0.23 nM T89988 CIKD64 44425653 IC50 = 3.5 nM T89988 CVW1F0 44425654 IC50 = 67 nM T89988 CT93GC 44439155 IC50 = 185 nM T89988 C58AVC 44439156 IC50 = 2840 nM T89988 CNW2K9 44439157 IC50 = 9332 nM T89988 CS5YO0 44439158 IC50 = 1123 nM T89988 C8GKW0 44439159 IC50 = 1803 nM T89988 CF6KR3 44439160 IC50 = 4741 nM T89988 CN7KQ2 44439163 IC50 = 118 nM T89988 C8QRF1 44439164 IC50 = 7601 nM T89988 CXNE20 44439166 IC50 = 43 nM T89988 C01KCX 44439169 IC50 = 106.91 nM T89988 C6PS5Z 44439170 IC50 = 52 nM T89988 CGYJ76 44439173 IC50 = 6475 nM T89988 CUT9L0 44441347 IC50 = 10 nM T89988 CAG6R0 44441352 IC50 = 10 nM T89988 CBY68G 44441356 IC50 = 180 nM T89988 CB28GP 44441358 IC50 = 120 nM T89988 CDI1Z6 44441359 IC50 = 170 nM T89988 CT4L3X 44441382 IC50 = 2050 nM T89988 CJTZ15 44441396 IC50 = 290 nM T89988 C4Z6BD 44442531 IC50 = 560 nM T89988 C2AY8H 44442532 IC50 = 110 nM T89988 C4D7BR 44442540 IC50 = 15000 nM T89988 CN3AK1 44442541 IC50 = 22000 nM T89988 CR5UZ7 44442542 IC50 = 3000 nM T89988 CAIO38 44442543 IC50 = 410 nM T89988 CA37EK 44442544 IC50 = 770 nM T89988 CB8UD0 44442547 IC50 = 150 nM T89988 CPH7V8 44442553 IC50 = 130 nM T89988 CSN9R7 44442554 IC50 = 120 nM T89988 C6Z4LR 44442555 IC50 = 120 nM T89988 C45LKM 44442556 IC50 = 190 nM T89988 CGI4O8 44442557 IC50 = 100 nM T89988 CW2Q1E 44442558 IC50 = 99 nM T89988 CWR41K 44442559 IC50 = 150 nM T89988 C6JA2N 44442560 IC50 = 200 nM T89988 C7CZI3 44442561 IC50 = 60 nM T89988 C1ASE4 44442562 IC50 = 260 nM T89988 CDNB78 44442563 IC50 = 490 nM T89988 CUNH60 44442564 IC50 = 750 nM T89988 CSK0B1 44442565 IC50 = 400 nM T89988 CDX9K1 44442566 IC50 = 380 nM T89988 CSRO45 44442569 IC50 = 7200 nM T89988 C3R4SV 44442570 IC50 = 1700 nM T89988 C1AK7V 44442571 IC50 = 1100 nM T89988 C98JQT 44442572 IC50 = 530 nM T89988 C3E8MO 44442573 IC50 = 430 nM T89988 CM62RJ 44442574 IC50 = 900 nM T89988 CB1D2L 44442575 IC50 = 160 nM T89988 CZ1Q3R 44442576 IC50 = 47 nM T89988 C23KHI 44442577 IC50 = 36 nM T89988 CX2U4T 44442578 IC50 = 36 nM T89988 CHA6Z3 44442580 IC50 = 670 nM T89988 CTE0Y1 44442581 IC50 = 120 nM T89988 CVC6E9 44442582 IC50 = 690 nM T89988 CHD74R 44442583 IC50 = 1300 nM T89988 C6F9PC 44442584 IC50 = 5600 nM T89988 CWCY76 44442586 IC50 = 720 nM T89988 C89VZB 44442587 IC50 = 39 nM T89988 C6W0XY 44442588 IC50 = 23 nM T89988 CD50ZB 44442589 IC50 = 65 nM T89988 C6M2TZ 44442590 IC50 = 240 nM T89988 C5Q7BK 44442591 IC50 = 90 nM T89988 C0GN4C 44442592 IC50 = 16 nM T89988 C93GZU 44442593 IC50 = 19 nM T89988 CRB1M8 44442594 IC50 = 110 nM T89988 C2B8QU 44442595 IC50 = 130 nM T89988 CO1F2A 44442596 IC50 = 310 nM T89988 CU43VX 44442598 IC50 = 37 nM T89988 C84AZN 44442599 IC50 = 20 nM T89988 CG8MC4 44443989 IC50 = 3100 nM T89988 C8TB1M 44443996 IC50 = 2900 nM T89988 CW9ML2 44444000 IC50 = 4500 nM T89988 CGN73S 44444001 IC50 = 1900 nM T89988 COJ91E 44444002 IC50 = 2300 nM T89988 CLW9O7 44444003 IC50 = 2600 nM T89988 C3G4RP 44444005 IC50 = 3800 nM T89988 CC50LS 44444006 IC50 = 3400 nM T89988 C8P6IQ 44444007 IC50 = 1800 nM T89988 C94CZJ 44444008 IC50 = 1200 nM T89988 C18RYD 44444009 IC50 = 2100 nM T89988 C3UJV4 44444032 IC50 = 1500 nM T89988 CI7ZK4 44444035 IC50 = 12600 nM T89988 C2NU7P 44444096 IC50 = 11100 nM T89988 CWB08Z 44444098 IC50 = 4000 nM T89988 CD82NB 44444099 IC50 = 320 nM T89988 CB9HW7 44444100 IC50 = 950 nM T89988 C2N9YB 44444102 IC50 = 510 nM T89988 CQ2U7T 44444103 IC50 = 2200 nM T89988 CJY6E1 44444104 IC50 = 2000 nM T89988 C9WUP6 44444105 IC50 = 5900 nM T89988 C27YJV 44444106 IC50 = 1400 nM T89988 C7I1MY 44444107 IC50 = 5200 nM T89988 C9R3XK 44444109 IC50 = 2900 nM T89988 CLV8O7 44444110 IC50 = 140 nM T89988 C2O0GB 44444111 IC50 = 180 nM T89988 CU7I5F 44444112 IC50 = 240 nM T89988 C8T6RW 44444113 IC50 = 130 nM T89988 C3VNH1 44444114 IC50 = 790 nM T89988 C98NMR 44446951 Ki = 1700 nM T89988 COP46Z 44447424 IC50 = 229.09 nM T89988 CW1Q8I 44447426 IC50 = 193 nM T89988 C4Y9JZ 44447427 IC50 = 204.17 nM T89988 COPZ27 44447429 IC50 = 14 nM T89988 CY5CA3 44447431 IC50 = 28.18 nM T89988 C0YB3Q 44447432 IC50 = 25.12 nM T89988 C0F8BO 44447433 IC50 = 281.84 nM T89988 C93BDA 44447434 IC50 = 285 nM T89988 CQ1PG4 44447435 IC50 = 125.89 nM T89988 CB9UO3 44447436 IC50 = 642 nM T89988 C49XWQ 44447446 IC50 = 229.09 nM T89988 CI8Q9M 44447766 IC50 = 3 nM T89988 C50JFH 44447775 IC50 = 4 nM T89988 CWY54R 44447782 IC50 = 6 nM T89988 C2UGM9 44447783 IC50 = 6 nM T89988 CSLU08 44447786 IC50 = 41 nM T89988 CRV6F7 44447789 IC50 = 45 nM T89988 CDI1F4 44447815 IC50 = 24 nM T89988 CMR4P3 44448776 IC50 = 50 nM T89988 CD3K4H 44448807 IC50 = 10 nM T89988 C12TPU 44448839 IC50 = 1 nM T89988 CB7F4C 44448879 IC50 = 1 nM T89988 CNPS37 44448915 IC50 = 2 nM T89988 C3UN9M 44448948 IC50 = 20 nM T89988 CUG0K5 44449030 IC50 = 20 nM T89988 CUV2A8 44449031 IC50 = 30 nM T89988 CV5G3U 44449054 IC50 = 2 nM T89988 C3NAM2 44449081 IC50 = 9 nM T89988 CIV30A 44449174 IC50 = 20 nM T89988 CU6M8T 44449175 IC50 = 80 nM T89988 CLB90E 44449204 IC50 = 2400 nM T89988 C6Q8HS 44449229 IC50 = 4800 nM T89988 CF5B8G 44453002 IC50 = 10000 nM T89988 CF0EB1 44453004 IC50 = 22000 nM T89988 C72NCT 44453133 IC50 > 10000 nM T89988 CEGW75 44453134 IC50 = 489 nM T89988 C9GNP8 44453171 IC50 = 473 nM T89988 C7PH5L 44453173 IC50 > 10000 nM T89988 CA0MZ6 44453203 IC50 > 5000 nM T89988 CALV41 44453204 IC50 > 5000 nM T89988 CSXO73 44453208 IC50 = 10000 nM T89988 C6G5AC 44453234 IC50 = 103 nM T89988 CESK25 44453268 IC50 = 305 nM T89988 C46MAN 44453298 IC50 = 5.5 nM T89988 C4ESA8 44453300 IC50 = 21 nM T89988 CH6C5F 44453325 IC50 = 53 nM T89988 CFH6C8 44453327 EC50 = 20 nM T89988 C0DM8U 44453329 IC50 = 121 nM T89988 C6M7IQ 44453330 IC50 = 21 nM T89988 CJV36D 44453365 IC50 = 5.3 nM T89988 CBNQ71 44453366 IC50 = 14 nM T89988 C2U5JW 44453368 IC50 = 6.1 nM T89988 C2JQ0A 44453369 IC50 = 2400 nM T89988 CI0PV7 44453370 IC50 = 2380 nM T89988 CV1E8J 44453372 IC50 = 59 nM T89988 CBCW46 44453373 IC50 = 35 nM T89988 CVC27Y 44453405 IC50 = 11 nM T89988 C1I9TO 44453407 IC50 = 20 nM T89988 CF8D2E 44453408 IC50 = 5.1 nM T89988 CE8X3Z 44453409 IC50 = 116 nM T89988 CBT74X 44453440 IC50 = 0.89 nM T89988 C9QKA4 44453441 IC50 = 116 nM T89988 CVL1R5 44453442 IC50 = 20 nM T89988 C06ICO 44453443 IC50 > 10000 nM T89988 CM9U2O 44453444 IC50 > 10000 nM T89988 C9Q1SV 44453471 IC50 = 43 nM T89988 CKX1I6 44453472 IC50 = 26 nM T89988 C3U2MW 44453473 IC50 = 643 nM T89988 CNT1L8 44453474 IC50 = 22 nM T89988 CPY9T6 44453475 IC50 > 10000 nM T89988 CY48QG 44453476 IC50 > 10000 nM T89988 CMBQ96 44453477 IC50 = 3100 nM T89988 C72HIV 44453505 IC50 > 5000 nM T89988 CEL4U0 44453507 IC50 = 74 nM T89988 CRZV62 44453533 IC50 = 730 nM T89988 CQ57XT 44453534 IC50 = 77 nM T89988 C2O5UN 44453535 IC50 = 300 nM T89988 CG0S3F 44453536 IC50 = 1360 nM T89988 C9X0RM 44453538 IC50 = 127 nM T89988 C8ZC4N 44453562 IC50 = 43 nM T89988 CBG8E7 44453563 IC50 = 2650 nM T89988 CMT4A6 44453565 IC50 = 630 nM T89988 CV85SI 44453587 IC50 > 10000 nM T89988 COK3C9 44453592 IC50 = 418 nM T89988 CWG31M 44453620 IC50 = 1550 nM T89988 C8ZA9E 44453621 IC50 > 10000 nM T89988 CY4ML1 44454793 IC50 = 115 nM T89988 CS2G0H 44454820 IC50 = 1.4 nM T89988 CT5N4E 44555481 IC50 > 50000 nM T89988 CQU5N6 44563038 IC50 = 1900 nM T89988 CR71SV 44563039 IC50 = 1300 nM T89988 CSQ4N3 44563071 IC50 = 960 nM T89988 CV2D1L 44563113 IC50 = 14 nM T89988 C5HIE4 44570713 IC50 = 112 nM T89988 C0OD7H 44570714 IC50 = 2 nM T89988 CQO26H 44570717 IC50 = 27 nM T89988 CF2N3O 44570718 IC50 = 7.7 nM T89988 C7ZYG6 44570779 IC50 = 135.7 nM T89988 C82AOH 44570780 IC50 = 227.5 nM T89988 CF56CE 44570781 IC50 = 23 nM T89988 CHB9E1 44571216 IC50 = 600 nM T89988 C2VC9W 44571218 IC50 = 4.8 nM T89988 CM4LZ8 44571257 IC50 = 19 nM T89988 CYCF52 44571258 IC50 = 61.5 nM T89988 C2OGV6 44573409 IC50 = 193.2 nM T89988 CZ4H9K 44573410 IC50 = 362 nM T89988 CGVT58 44573411 IC50 = 155.96 nM T89988 CYK18E 44573412 IC50 = 63.97 nM T89988 C09CJU 44573450 IC50 = 174.98 nM T89988 CKRY49 44573451 IC50 = 84.92 nM T89988 C6Z7DI 44573452 IC50 = 4.603 nM T89988 C3AG9N 44573485 IC50 = 4.6 nM T89988 C5OZX4 44573486 IC50 = 29.99 nM T89988 CR3XS9 44573487 IC50 = 35.97 nM T89988 C9FOB2 44573488 IC50 = 21.98 nM T89988 C9UH5E 44573535 IC50 = 630.96 nM T89988 CW7B8R 44573537 IC50 = 187 nM T89988 CO0FB9 44573538 IC50 = 187.07 nM T89988 CP9HC7 44573568 Ki = 50 nM T89988 C10UVI 44573569 IC50 = 418.79 nM T89988 C3RTY1 44573608 IC50 = 2.999 nM T89988 CWXH83 44573609 IC50 = 51 nM T89988 CBQ3N6 44573649 IC50 = 5.998 nM T89988 CCKN12 44573650 IC50 = 5.495 nM T89988 CYIP03 44573651 IC50 = 27.99 nM T89988 CQ2CP1 44573699 IC50 = 7 nM T89988 CBL9R6 44580424 IC50 = 1180 nM T89988 CD2V0I 44580590 IC50 = 4.3 nM T89988 C6MG8Q 44580591 IC50 = 6 nM T89988 CK78AN 44583280 IC50 = 24 nM T89988 CT78IF 44583281 IC50 = 6.5 nM T89988 CQI80O 44583282 IC50 = 16 nM T89988 C9KAN6 44583283 IC50 = 2.3 nM T89988 C8MIP6 44593554 IC50 = 1605 nM T89988 CTY83R 44593555 IC50 = 2 nM T89988 C9F8IU 44593561 IC50 = 3.3 nM T89988 C71ENV 44593562 IC50 = 238.78 nM T89988 CBR46V 44593563 IC50 = 0.3 nM T89988 CU7R2S 44593564 IC50 = 0.8 nM T89988 CSW0N7 44595711 IC50 = 11 nM T89988 C5IMW6 44612589 IC50 = 4500 nM T89988 C4D8RG 44612590 IC50 = 36 nM T89988 CU3C8Z 44612708 IC50 = 5779 nM T89988 CK3N1G 46206137 IC50 > 10000 nM T89988 CY2A9C 46240380 IC50 = 310 nM T89988 CIG71O 46240381 IC50 = 2700 nM T89988 CFY3L5 46240481 IC50 = 650 nM T89988 CPHB87 46240482 IC50 = 13 nM T89988 C8R1QX 46240484 IC50 = 60 nM T89988 CR0NX3 46240582 IC50 = 5300 nM T89988 CF9O5C 46240584 IC50 = 28 nM T89988 CV2X5E 46240585 IC50 = 70 nM T89988 CD1M3J 46240687 IC50 = 41 nM T89988 C63QWF 46240785 IC50 = 65 nM T89988 C3YU2T 46240895 IC50 = 36 nM T89988 CEH6U9 46241010 IC50 = 4 nM T89988 C43MLP 46241011 IC50 = 790 nM T89988 CJ7L3Z 46241120 IC50 = 100 nM T89988 C7PVU1 46241121 IC50 = 2820 nM T89988 CDZ3V6 46241509 IC50 = 56 nM T89988 CH8F5U 46241608 IC50 = 50 nM T89988 CD1H3B 46241609 IC50 = 250 nM T89988 CXJ7C5 46241610 IC50 = 17 nM T89988 C35CXM 46241611 IC50 = 71 nM T89988 C5Y8ZT 46241717 IC50 = 18 nM T89988 C8EX9T 46241718 IC50 = 43 nM T89988 CZK4H8 46241719 IC50 = 190 nM T89988 CK9H6B 46241720 IC50 = 170 nM T89988 CA05ZH 46241826 IC50 = 45 nM T89988 C3LD6V 46241827 IC50 = 220 nM T89988 CRJD47 46241829 IC50 = 190 nM T89988 C5TC2S 46830335 IC50 = 1.7 nM T89988 C1K7FL 46830336 IC50 = 3040 nM T89988 C5ZJM9 46842084 IC50 = 520 nM T89988 CPQ5E8 46842085 IC50 = 1730 nM T89988 C4Q6JH 46842086 IC50 = 750 nM T89988 CNX7H4 46842232 IC50 = 620 nM T89988 CU5W3P 46842233 IC50 = 3160 nM T89988 C5Y6MQ 46842235 IC50 = 660 nM T89988 CF8LO6 46842236 IC50 = 7520 nM T89988 CJDG46 46842381 IC50 = 1740 nM T89988 C2FE9H 46842382 IC50 = 6600 nM T89988 C1N4KX 46842383 IC50 = 580 nM T89988 CQN2H4 46865774 IC50 = 0.8 nM T89988 CPV2L4 46865775 IC50 = 0.5 nM T89988 CB8GE1 46884818 IC50 = 29 nM T89988 CHS4Q3 46884855 IC50 = 160 nM T89988 C4MQ0A 46884856 IC50 = 11 nM T89988 CCNT25 46884898 IC50 = 9 nM T89988 C3MSG2 46885027 IC50 = 9 nM T89988 CI5J4L 46885028 IC50 = 120 nM T89988 CA5W3K 46885029 IC50 = 170 nM T89988 C6QBR9 46885159 IC50 = 110 nM T89988 CMI8G7 46885160 IC50 = 1100 nM T89988 CB7XI0 46885213 IC50 = 2.6 nM T89988 CQ0M2Z 46885214 IC50 = 710 nM T89988 CB60AL 46885269 IC50 = 1860 nM T89988 C2VSQ4 46885270 IC50 > 10000 nM T89988 CLBQ50 46885271 IC50 > 10000 nM T89988 C1Z5OS 46886055 IC50 = 0.3 nM T89988 C7JO8A 46886056 IC50 = 51 nM T89988 CF83SA 46886057 IC50 = 4500 nM T89988 CA18BC 46886058 IC50 > 1000 nM T89988 CJ2U1P 46886059 IC50 = 284 nM T89988 C9QE0J 46886060 IC50 > 1000 nM T89988 CU9PR6 46886061 IC50 = 99 nM T89988 CNDL30 46886482 IC50 = 50 nM T89988 CTQ13P 46886507 IC50 = 311.5 nM T89988 C32NJX 46886508 IC50 = 278 nM T89988 CF8N0U 46886536 IC50 = 0.4 nM T89988 CZ59HO 46886537 IC50 = 151 nM T89988 C28IHA 46886538 IC50 = 3.5 nM T89988 C0UDN9 46886539 IC50 = 0.8 nM T89988 CK9E8N 46927116 IC50 = 36 nM T89988 C82HXR 46927117 IC50 = 7 nM T89988 CV28ZU 46944853 IC50 = 25 nM T89988 CT9P5G 46944854 IC50 = 32 nM T89988 CWH4K6 46944855 IC50 = 57 nM T89988 CC3O0S 46945254 IC50 = 35 nM T89988 C1UB8E 46945255 IC50 = 85 nM T89988 C4RZG5 46945857 IC50 = 44 nM T89988 CAK5J0 46946058 IC50 = 31 nM T89988 CY09UB 46946452 IC50 < 1000 nM T89988 CFH87K 46947816 IC50 = 13 nM T89988 CVEF51 49763568 IC50 = 5 nM T89988 C43LAE 49763569 IC50 = 390 nM T89988 CI6AR9 49763571 IC50 = 35 nM T89988 C78ICP 49763574 IC50 = 110 nM T89988 C65RMG 49763575 IC50 = 160 nM T89988 CQLN97 49763682 IC50 = 25 nM T89988 CY5ME3 49763685 IC50 = 80 nM T89988 C0ADU9 49763686 IC50 = 70 nM T89988 C1GVM0 49763804 IC50 = 61 nM T89988 C94ARN 49763931 IC50 = 21 nM T89988 C68SFM 49764196 IC50 = 22 nM T89988 CSW83Q 49764322 IC50 = 20 nM T89988 C1Z0UD 49764446 IC50 = 15 nM T89988 C5AD0E 49764447 IC50 = 21 nM T89988 C20WNR 49764700 IC50 = 210 nM T89988 CIZ86P 49764701 IC50 = 410 nM T89988 C95CPY 49798264 Ki = 251.19 nM T89988 C3SUN1 49798265 Ki = 31.62 nM T89988 CBG4T2 49798289 Ki = 125.89 nM T89988 C4HO3X 49798290 Ki > 3162.28 nM T89988 CK92RZ 49798291 Ki = 63.1 nM T89988 C70BOA 49798292 Ki = 39.81 nM T89988 C5LZJ7 49798323 Ki = 19.95 nM T89988 CX90YD 49798324 Ki > 3162.28 nM T89988 C8D3SA 49798325 Ki = 398.11 nM T89988 CMZT82 49798326 Ki = 630.96 nM T89988 CVD31B 49798327 Ki > 3162.28 nM T89988 CC42TS 49798347 Ki = 158.49 nM T89988 C4T3JR 49798348 Ki = 7.943 nM T89988 CQVG17 49798349 Ki = 3.162 nM T89988 C38JTB 49798350 Ki = 5.012 nM T89988 C94JQY 49798351 Ki = 398.11 nM T89988 C1WOS7 49798396 Ki = 794.33 nM T89988 CLD0Y3 49798397 Ki = 398.11 nM T89988 C3OMN2 49798398 Ki = 50.12 nM T89988 CG35HZ 49798399 Ki = 31.62 nM T89988 C3IDX4 49798434 Ki = 1.995 nM T89988 CQN90U 49798435 Ki = 1.585 nM T89988 CVG78D 49798436 Ki = 3.162 nM T89988 C62VRQ 49798437 Ki = 25.12 nM T89988 CR4FE3 49798438 Ki = 19.95 nM T89988 CY90CD 49798461 Ki = 10 nM T89988 CF8J6E 49798462 Ki = 12.59 nM T89988 C60QIU 49798463 Ki = 15.85 nM T89988 CD20QY 49798464 Ki = 199.53 nM T89988 CQP1H6 49798489 Ki = 50.12 nM T89988 CG42MY 49863167 IC50 = 2837.92 nM T89988 C9YB8V 49863168 IC50 = 9332.54 nM T89988 C41FAQ 49863199 IC50 = 1122.02 nM T89988 CTM2W6 49863200 IC50 = 1803.02 nM T89988 CQIV05 49863201 IC50 = 1224.62 nM T89988 C4SMG0 49863202 IC50 = 107.89 nM T89988 C6AP0W 49863225 IC50 = 42.95 nM T89988 C7JB8Z 50925394 IC50 = 0.95 nM T89988 C2T4IC 50991056 IC50 = 7.7 nM T89988 CI32TR 50992246 IC50 = 3 nM T89988 C8ICA4 51353692 IC50 > 10000 nM T89988 C4B0AF 51353693 IC50 > 10000 nM T89988 CX6B8U 52941377 IC50 = 2.9 nM T89988 CIBA52 52942863 IC50 = 120 nM T89988 C71MDG 52943756 IC50 = 7.4 nM T89988 CRKC87 52944966 IC50 = 17 nM T89988 CTF7Y6 52946110 IC50 > 1000 nM T89988 CRDI09 52947358 IC50 > 1000 nM T89988 CB4MN2 52947389 IC50 > 1000 nM T89988 CF9BQ7 52947417 IC50 = 649 nM T89988 CUFX45 52950180 IC50 = 47 nM T89988 CK0M6N 53317027 IC50 = 5 nM T89988 CT58US 53317028 IC50 = 3.2 nM T89988 C8BSM2 53317041 IC50 = 3.1 nM T89988 C8HO9F 53317526 IC50 = 221 nM T89988 CCN50W 53317527 IC50 = 232 nM T89988 C6FG7U 53318314 IC50 = 11.6 nM T89988 C5MFO3 53318315 IC50 = 13 nM T89988 C2PK1V 53318316 IC50 = 4.2 nM T89988 C0AS8E 53318853 IC50 = 2.5 nM T89988 C8K5QI 53318854 IC50 = 46.5 nM T89988 C1GH4U 53318855 IC50 = 116 nM T89988 C0VGT5 53319664 IC50 = 11.1 nM T89988 CZU3G0 53320171 IC50 = 22.7 nM T89988 CS2QA6 53320349 IC50 = 32 nM T89988 CI0R1F 53320350 IC50 = 17 nM T89988 CI2JU6 53320967 IC50 = 36.9 nM T89988 C1NAP2 53320968 IC50 = 130 nM T89988 CL0SO8 53320970 IC50 = 38.4 nM T89988 CNQ30U 53320973 IC50 = 4.3 nM T89988 C57FLU 53320974 IC50 = 75.9 nM T89988 C76HPL 53321427 IC50 = 45.5 nM T89988 C1HOS5 53321482 IC50 = 11.5 nM T89988 CW1TY6 53321483 IC50 = 10.6 nM T89988 C17BAO 53321484 IC50 = 27.6 nM T89988 CTHX71 53321503 IC50 = 18.5 nM T89988 CBJR38 53321615 IC50 = 39.5 nM T89988 CK2M9J 53321616 IC50 = 2.3 nM T89988 CFW3C6 53322299 IC50 = 14.6 nM T89988 CK2JD6 53322809 IC50 = 5.7 nM T89988 C35XLW 53322810 IC50 = 8.5 nM T89988 C8VM2O 53322811 IC50 = 9.3 nM T89988 C5BPW8 53322812 IC50 = 19.5 nM T89988 CYK8U9 53322813 IC50 = 294 nM T89988 C3JDS8 53322831 IC50 > 1000 nM T89988 CH6MZ9 53323653 IC50 = 3.5 nM T89988 C5J2DH 53323654 IC50 = 11.7 nM T89988 C3WY6T 53323664 IC50 = 15.2 nM T89988 CH3LK8 53324139 IC50 = 175 nM T89988 COYC36 53324140 IC50 = 46 nM T89988 C48XCJ 53324141 IC50 = 66 nM T89988 CO93PA 53324304 IC50 = 7 nM T89988 C09CEX 53324942 IC50 = 6.5 nM T89988 CHW4E1 53324943 IC50 = 12.8 nM T89988 CF93PO 53324944 IC50 = 17.5 nM T89988 C9YGA3 53325385 IC50 = 28 nM T89988 CM12CJ 53325460 IC50 = 3.2 nM T89988 CY15EU 53325639 IC50 = 6.2 nM T89988 CV4AO0 53326225 IC50 = 12.2 nM T89988 CU17IJ 53326226 IC50 = 14.7 nM T89988 C4N1PX 53326242 IC50 = 28 nM T89988 CHX40S 53326386 IC50 = 2.9 nM T89988 C5NS6A 53326645 IC50 = 17.3 nM T89988 CD1SK7 53326700 IC50 = 462 nM T89988 C8E0DF 53326701 IC50 = 15 nM T89988 C7PQ1Y 53326702 IC50 = 36 nM T89988 CRF7T6 53326703 IC50 = 34 nM T89988 CYH0F6 53326721 IC50 = 17 nM T89988 C2S5ZK 53326900 IC50 = 251 nM T89988 C6KP2D 53326901 IC50 = 13.9 nM T89988 CIT7E8 53389636 Ki = 3.467 nM T89988 CC8ME1 53389637 Ki = 1.9 nM T89988 CAH13N 53389641 Ki = 3.981 nM T89988 CM4U5G 53389660 Ki = 1.7 nM T89988 C13SIB 53389710 Ki = 2.291 nM T89988 CXW05M 53389845 Ki = 1.259 nM T89988 CS0Q8N 53389902 Ki = 0.4 nM T89988 C8GNX3 53389980 Ki = 16.6 nM T89988 C4AKQ1 54580188 IC50 = 18.3 nM T89988 CC72WM 54580189 IC50 = 68.6 nM T89988 C89MEB 54580190 IC50 = 15.5 nM T89988 CC3J5L 54581190 IC50 = 43.7 nM T89988 CG3HB9 54582215 IC50 = 40.1 nM T89988 C4KMX1 54582216 IC50 = 29.1 nM T89988 CD1AE2 54582217 IC50 = 20.9 nM T89988 CLX7U9 54583111 IC50 = 4.5 nM T89988 C3WZ9I 54583112 IC50 = 31.9 nM T89988 CYD20W 54583185 IC50 = 17.8 nM T89988 COQD25 54583186 IC50 = 9.2 nM T89988 CC19ZA 54583187 IC50 = 15.4 nM T89988 C9GFR1 54584109 IC50 = 500 nM T89988 C90AHI 54584164 IC50 = 28 nM T89988 CZ4S0B 54585107 IC50 = 18.3 nM T89988 C3TAR4 54585108 IC50 = 71.5 nM T89988 C8RTU2 54585109 IC50 = 19.7 nM T89988 CC6HY7 54586021 IC50 = 9.5 nM T89988 C7V0YA 54597147 Ki = 15 nM T89988 CGIP16 54754722 IC50 = 47 nM T89988 CX4LK5 54754723 IC50 = 86 nM T89988 C6LZ8B 54754724 IC50 = 32 nM T89988 CSA9I6 54754844 IC50 = 330 nM T89988 CEGJ53 54754845 IC50 = 510 nM T89988 C9NV8L 54754967 IC50 = 16 nM T89988 CI78YZ 54754968 IC50 = 2 nM T89988 CV3K8U 54754969 IC50 = 3 nM T89988 C6T8XS 54755079 IC50 = 12 nM T89988 CL2AU5 54755081 IC50 = 27 nM T89988 C2R6KO 54755083 IC50 = 63 nM T89988 C5LT0A 54755193 IC50 = 370 nM T89988 C3SD6W 54755560 IC50 = 7 nM T89988 C4GBT5 54755562 IC50 = 230 nM T89988 C0KZ4M 54755801 IC50 = 20 nM T89988 C2QP4W 54755919 IC50 = 20 nM T89988 CPWZ05 54756038 IC50 = 29 nM T89988 CJBW64 54756045 IC50 = 14 nM T89988 C0ZWL2 54756156 IC50 = 28 nM T89988 CFHI34 54768835 IC50 = 17 nM T89988 CLY35F 54768836 IC50 = 21 nM T89988 C9U4YQ 54768838 IC50 = 8 nM T89988 CO4FY1 54769305 IC50 = 15 nM T89988 CF39PC 54769752 IC50 = 19 nM T89988 CWN90Q 54771978 IC50 = 20 nM T89988 CUM4B5 54771980 IC50 = 5 nM T89988 CL7UD5 54772203 IC50 = 5 nM T89988 CH7K6J 54772204 IC50 = 7 nM T89988 C4E5YQ 54772205 IC50 = 7 nM T89988 C7Y8KR 54772206 IC50 = 7 nM T89988 C3UJ2D 56643545 IC50 = 4 nM T89988 C94RZF 56657929 IC50 = 19 nM T89988 COST81 56657930 IC50 = 4 nM T89988 C21NEQ 56659196 IC50 = 29 nM T89988 C7B9TW 56659197 IC50 = 33 nM T89988 CUM53N 56659295 IC50 = 20 nM T89988 C4IZL5 56661444 IC50 = 55 nM T89988 CQ25TB 56661451 IC50 = 7 nM T89988 CC3XP8 56661559 IC50 = 2600 nM T89988 C7K4TJ 56662695 IC50 = 7 nM T89988 C7SJH2 56664979 IC50 = 8 nM T89988 CC5S6K 56667036 IC50 = 45 nM T89988 C4X5DR 56668306 IC50 = 290 nM T89988 CF2N5W 56668309 IC50 = 82 nM T89988 C4SP2W 56668313 IC50 = 650 nM T89988 C31SKP 56668413 IC50 > 25000 nM T89988 CI5Y4E 56669631 IC50 = 200 nM T89988 CKV58T 56670477 IC50 > 25000 nM T89988 C34WPT 56671792 IC50 = 30 nM T89988 CXUJ14 56671793 IC50 = 11 nM T89988 C4UHW2 56671794 IC50 = 9 nM T89988 CG1JX9 56671795 IC50 = 11 nM T89988 CXIQ98 56671923 IC50 = 9 nM T89988 C19LWV 56671924 IC50 = 120 nM T89988 CE3Y0C 56671925 IC50 = 13 nM T89988 CET7K4 56672021 IC50 = 10000 nM T89988 CY26SL 56675205 IC50 = 6 nM T89988 C03LOT 56675300 IC50 = 530 nM T89988 CK9JX5 56675301 IC50 = 140 nM T89988 CU0H6Z 56675302 IC50 = 200 nM T89988 CR51UE 56676473 IC50 = 1400 nM T89988 C0KG7I 56676474 IC50 = 27 nM T89988 CBTG12 56677288 IC50 = 25 nM T89988 CU35WX 56677289 IC50 > 25000 nM T89988 C1E9CF 56677290 IC50 > 25000 nM T89988 CV23WU 56677291 IC50 > 25000 nM T89988 CCV03M 56677295 IC50 > 25000 nM T89988 CE3T1U 56677296 IC50 = 1200 nM T89988 CR8ZJ4 56678497 IC50 = 510 nM T89988 CD8IZ5 56678506 IC50 = 920 nM T89988 C7QW5F 56678507 IC50 = 14 nM T89988 C7MXE5 56678508 IC50 = 17 nM T89988 C2O4SY 56678640 IC50 = 2080 nM T89988 CKAU07 56680600 IC50 = 1000 nM T89988 C1BI5O 56681842 IC50 = 5400 nM T89988 CIW1T6 56683044 IC50 = 29 nM T89988 CKVB12 56683116 IC50 = 5 nM T89988 C0ZH9W 56683120 IC50 = 480 nM T89988 C9KMN5 56683121 IC50 = 37 nM T89988 CNS7H5 57335017 IC50 = 6.6 nM T89988 C6OX7Y 57343820 IC50 = 130 nM T89988 C3ME6N 57344218 IC50 = 190 nM T89988 CN0U5G 57344221 IC50 = 490 nM T89988 C6EGO0 57344296 IC50 = 36 nM T89988 C1GZ6S 57344297 IC50 = 270 nM T89988 C23CNI 57344298 IC50 = 64 nM T89988 CT92GZ 57344299 IC50 = 140 nM T89988 CBW8S6 57344303 IC50 = 16 nM T89988 C3ADF6 57344305 IC50 = 35 nM T89988 C5GV0P 57344307 IC50 = 83 nM T89988 C73ZNA 57344310 IC50 = 130 nM T89988 C9YZU2 57344314 IC50 = 900 nM T89988 C6MI0E 57344315 IC50 = 640 nM T89988 CVO80U 57344316 IC50 = 670 nM T89988 C4UC8E 57344317 IC50 = 980 nM T89988 CH7NM1 57344318 IC50 = 980 nM T89988 CI61XO 57391449 Ki = 40 nM T89988 CU39WF 57391450 Ki = 200 nM T89988 CW5GM2 57391487 IC50 = 950 nM T89988 CZOY39 57391591 IC50 = 6.6 nM T89988 CBEO41 57391765 IC50 = 7.3 nM T89988 CK9L1O 57391766 IC50 = 10.9 nM T89988 CN1Q4Y 57391767 IC50 = 2.7 nM T89988 CC53ND 57391768 IC50 = 7.8 nM T89988 CCZ85S 57391797 IC50 = 3700 nM T89988 CGR4B9 57392725 IC50 = 1878 nM T89988 CD97NH 57393218 Ki = 79 nM T89988 CF2WS8 57393219 Ki = 63 nM T89988 CRU9I7 57393220 Ki = 10 nM T89988 C3VI0X 57393248 IC50 > 25000 nM T89988 COE45G 57393249 IC50 = 740 nM T89988 C94QJG 57393347 IC50 = 12 nM T89988 CV4F2A 57393495 Ki = 63 nM T89988 C60XVA 57393496 Ki = 25 nM T89988 CW93MJ 57393497 Ki = 25 nM T89988 CHN9C0 57393530 IC50 = 59 nM T89988 CQW74A 57393531 IC50 = 310 nM T89988 CKJX42 57394938 Ki = 100 nM T89988 CA08MX 57394939 Ki = 631 nM T89988 CLFR28 57394966 IC50 = 25000 nM T89988 C4Y7BS 57394967 IC50 = 8600 nM T89988 CR37GS 57394968 IC50 = 9200 nM T89988 CY4JZ1 57394969 IC50 = 6000 nM T89988 C39SHX 57394970 IC50 = 15800 nM T89988 CC14HJ 57394971 IC50 > 25000 nM T89988 C7OF3Z 57395061 IC50 = 370 nM T89988 C3QCD9 57395216 IC50 = 9.3 nM T89988 C94MZO 57395217 IC50 = 3.2 nM T89988 CDIF34 57395218 IC50 = 2.6 nM T89988 C81ASJ 57395219 IC50 = 3 nM T89988 CD6F3G 57395221 Ki = 8 nM T89988 CKTL37 57396690 Ki = 794 nM T89988 CV9RJ7 57396722 IC50 = 5200 nM T89988 C7JOW2 57396723 IC50 = 2300 nM T89988 C5ZGD3 57396724 IC50 = 1300 nM T89988 CDY14H 57396725 IC50 = 1300 nM T89988 C6NPG0 57396726 IC50 = 11600 nM T89988 C0D3HL 57396832 IC50 = 130 nM T89988 CXB1F0 57396900 IC50 = 72 nM T89988 CH3CT2 57396901 IC50 = 27 nM T89988 CV4CN3 57396998 IC50 = 14 nM T89988 CO37CB 57396999 IC50 = 2.4 nM T89988 C5CYT8 57397001 Ki = 8 nM T89988 C7CHF8 57397013 IC50 = 4100 nM T89988 C9HF6A 57398458 Ki = 10 nM T89988 CK4E3W 57398492 IC50 > 25000 nM T89988 C3W1JY 57398493 IC50 = 9572 nM T89988 CO3UM0 57398494 IC50 = 1890 nM T89988 CQS9E4 57398590 IC50 = 340 nM T89988 CX8N3C 57398651 IC50 = 570 nM T89988 CYO6T8 57398750 IC50 = 4.9 nM T89988 CVF50W 57400125 Ki = 13 nM T89988 CH1KQ9 57400126 Ki = 13 nM T89988 CR09LY 57400127 Ki = 3 nM T89988 C6V8ET 57400128 Ki = 16 nM T89988 CNHU38 57400129 Ki = 2 nM T89988 C27JYV 57400160 IC50 = 50 nM T89988 CZ41PU 57400161 IC50 = 8100 nM T89988 CJ5X8T 57400162 IC50 > 25000 nM T89988 CV42YH 57400331 IC50 = 34 nM T89988 CWR51A 57400420 Ki = 4 nM T89988 C4O0ML 57400451 IC50 = 5.2 nM T89988 C2YVE5 57400452 IC50 = 12 nM T89988 C1N8YX 57401421 IC50 = 925 nM T89988 C67VKS 57401953 IC50 > 25000 nM T89988 C9SZ0F 57401954 IC50 = 38 nM T89988 CR6D1J 57402059 IC50 = 89 nM T89988 C2XM3P 57402124 IC50 = 180 nM T89988 CV54BI 57402219 IC50 = 1 nM T89988 CQ3JU8 57402220 IC50 > 1000 nM T89988 CE9TB4 57402254 IC50 = 2900 nM T89988 C5LG7S 57403699 IC50 = 2200 nM T89988 C8XIR4 57403700 IC50 = 1400 nM T89988 CG5X8H 57403701 IC50 > 25000 nM T89988 C5GI7L 57403755 IC50 > 25000 nM T89988 CRSG52 57403811 IC50 = 34 nM T89988 CJ2K4V 57403877 IC50 = 54 nM T89988 CM32RA 57656640 IC50 = 27 nM T89988 C0OJA5 57656641 IC50 = 17 nM T89988 CT8V9X 57656657 IC50 = 31 nM T89988 CH7BO0 57656701 IC50 = 5500 nM T89988 CMI4T3 57656713 IC50 = 64 nM T89988 CB30PQ 57656715 IC50 = 64 nM T89988 C51DOT 57656719 IC50 = 68 nM T89988 C2GHC7 57656729 IC50 = 2570 nM T89988 C6W3EJ 57656749 IC50 = 421 nM T89988 C1KAC6 57656808 IC50 = 797 nM T89988 CN7O1T 57656825 IC50 = 75 nM T89988 CHJ87A 57656833 IC50 = 3.5 nM T89988 CS6O1V 57656854 IC50 = 32 nM T89988 CPN5S4 57656869 IC50 = 262 nM T89988 CU8I2F 57656871 IC50 = 21 nM T89988 CD5W4E 57656887 IC50 = 202 nM T89988 C7NF4J 57656915 IC50 = 710 nM T89988 CQX1D5 57656921 IC50 = 58 nM T89988 C1QSF4 57656938 IC50 = 98 nM T89988 C5V0JI 57656942 IC50 = 220 nM T89988 C0YWT1 58509213 IC50 > 10000 nM T89988 CWFC53 59370257 IC50 = 0.65 nM T89988 CEB7T9 59370267 IC50 < 0.45 nM T89988 CN0C8R 60148505 IC50 = 6.5 nM T89988 CQR25M 66767933 IC50 < 0.45 nM T89988 CO62SG 66768099 IC50 < 0.45 nM T89988 CC81NU 66768640 IC50 = 4.9 nM T89988 C85HLV 67011331 IC50 = 3.4 nM T89988 C7CDA0 67220645 IC50 = 69 nM T89988 CC28AD 68003782 IC50 = 22 nM T89988 CXU2T6 68003962 IC50 = 15 nM T89988 C7ZA5Y 68003997 IC50 = 23 nM T89988 CQ4M8Y 68004002 IC50 = 40 nM T89988 CB7T0X 68004010 IC50 = 22 nM T89988 C9SZT4 68004011 IC50 = 19 nM T89988 C9BFS2 68004012 IC50 = 27 nM T89988 CX0B4G 68004016 IC50 = 38 nM T89988 C6U9NR 68004034 IC50 = 10 nM T89988 C8EM6J 68004094 IC50 = 72 nM T89988 CCO4A2 68004146 IC50 = 56 nM T89988 CFX59N 68070944 Ki = 24 nM T89988 C4D5IO 68616341 IC50 = 28 nM T89988 CCB1T5 68764898 IC50 = 0.24 nM T89988 C5O0JN 68764925 IC50 = 0.5 nM T89988 C70QJS 68767049 IC50 = 0.6 nM T89988 C8VU1C 68767078 IC50 = 2.7 nM T89988 C8XT7M 68767109 IC50 = 5.2 nM T89988 CP23JT 68767124 IC50 = 1.2 nM T89988 CKWJ72 68767577 IC50 = 0.2 nM T89988 C8U1DK 68767802 IC50 = 0.7 nM T89988 CS7T1U 68768752 IC50 = 2.2 nM T89988 CRM71Y 68768923 IC50 = 1.3 nM T89988 C6L3ZT 68769143 IC50 = 0.6 nM T89988 CHS3Z2 68769744 IC50 = 0.5 nM T89988 C2YRL3 68769802 IC50 = 3 nM T89988 C39SPK 68772423 IC50 = 0.9 nM T89988 C1UMP9 68867935 IC50 = 1.1 nM T89988 CWZU52 68988296 IC50 = 0.96 nM T89988 C5MP1I 69035439 IC50 = 1.2 nM T89988 CIU35O 69035677 IC50 = 1.9 nM T89988 C9UI0T 69212799 EC50 = 360 nM T89988 CPGC67 69285465 IC50 = 20 nM T89988 CM5XA1 69285531 IC50 = 13 nM T89988 C0QZ4U 69285563 IC50 = 33 nM T89988 C5T2GC 69285794 IC50 = 2.5 nM T89988 C8R4LZ 69286108 IC50 = 41 nM T89988 CNT95I 69286635 IC50 = 4.7 nM T89988 C1NY8Q 69315675 IC50 = 1700 nM T89988 C46QLW 69321774 IC50 = 440 nM T89988 CAU52S 70681271 IC50 = 158 nM T89988 C2K5HI 70681778 IC50 = 1055 nM T89988 CRZ9P2 70681779 IC50 > 10000 nM T89988 C8VE1I 70683350 IC50 = 3.8 nM T89988 CA1W4H 70683355 IC50 = 28000 nM T89988 CVUR18 70683619 IC50 = 860 nM T89988 C45LTY 70686028 IC50 > 10000 nM T89988 CSA38W 70687885 IC50 = 35 nM T89988 C4CI2T 70687886 IC50 = 84 nM T89988 CIS85H 70688149 IC50 = 26 nM T89988 C5M1GF 70689909 IC50 = 18 nM T89988 C9RDP5 70689914 IC50 = 11 nM T89988 C0QUO1 70689915 IC50 = 3.3 nM T89988 C7ESZ0 70691783 IC50 = 180 nM T89988 CTDY17 70691784 IC50 = 5 nM T89988 CNSJ34 70691785 IC50 = 10 nM T89988 C2GXN6 70692344 IC50 = 780 nM T89988 C3G7YH 70693849 IC50 = 10 nM T89988 CG7U4L 70696469 IC50 = 1458 nM T89988 CXS70G 70696470 IC50 = 449 nM T89988 C35YZQ 70697571 EC50 = 810 nM T89988 C5GM9Y 71190126 IC50 = 5 nM T89988 CG3DM1 71214709 Ki = 10 nM T89988 CG5V6I 71214710 Ki = 15.85 nM T89988 CA72CU 71214725 Ki = 39.81 nM T89988 CMSH09 71214976 Ki = 12.59 nM T89988 CRSA04 71226374 IC50 = 125 nM T89988 CSD6R9 71450657 Ki = 25.12 nM T89988 C8A0XW 71450658 Ki = 10 nM T89988 CW6C9V 71452241 IC50 = 33 nM T89988 C8YW2L 71452487 Ki = 100 nM T89988 C1TOE8 71452488 Ki = 50.12 nM T89988 C71FXH 71454246 Ki = 501.19 nM T89988 CD8I7C 71454247 Ki = 100 nM T89988 CSL01M 71454248 Ki = 12.59 nM T89988 C3EYK5 71456007 Ki = 1584.89 nM T89988 CHV16Z 71456008 Ki = 63.1 nM T89988 C6MHX5 71457815 Ki = 50.12 nM T89988 C3BXS9 71461438 Ki = 10 nM T89988 CRV73F 71461439 Ki = 100 nM T89988 C3P5HM 71461440 Ki = 31.62 nM T89988 C5E1FJ 71463165 Ki = 1258.93 nM T89988 C8VX0L 71463166 Ki = 251.19 nM T89988 CPU23H 71517239 IC50 = 4070 nM T89988 CLAF67 71517240 IC50 = 23 nM T89988 CYSI71 71517241 IC50 = 150 nM T89988 C8SR2Q 71517242 IC50 = 20 nM T89988 C4TGH7 71517401 IC50 = 45 nM T89988 CU28ZL 71517402 IC50 = 1258 nM T89988 C0BWE4 71517403 IC50 = 263 nM T89988 CU2TR7 71517573 IC50 = 59 nM T89988 C1XWC3 71517574 IC50 = 58 nM T89988 CZ5QD8 71517575 IC50 = 210 nM T89988 CGE96J 71517576 IC50 = 200 nM T89988 CFZ27L 71517577 IC50 = 8095 nM T89988 CK81FA 71517737 IC50 = 247 nM T89988 CVN31I 71518405 IC50 = 3300 nM T89988 CTL9E5 71518406 IC50 = 2329 nM T89988 C9V5RD 71518407 IC50 = 1529 nM T89988 CW39SU 71518408 IC50 = 699 nM T89988 CH5UM0 71518570 IC50 = 874 nM T89988 C6DIG9 71518571 IC50 = 3558 nM T89988 CZ0S5X 71518572 IC50 > 25000 nM T89988 CEJ1O6 71518573 IC50 > 25000 nM T89988 CQC14H 71518574 IC50 = 76 nM T89988 CXV79I 71518727 IC50 = 7927 nM T89988 CMKZ52 71518728 IC50 = 1070 nM T89988 CL05CZ 71518896 IC50 > 25000 nM T89988 C4UMA0 71518897 IC50 = 1100 nM T89988 C3Y2CP 71518898 IC50 = 200 nM T89988 CGO9T8 71519050 IC50 = 1500 nM T89988 CSU8J9 71519051 IC50 > 25000 nM T89988 C0E9LJ 71519052 IC50 = 5600 nM T89988 CK1GR7 71519053 IC50 = 4400 nM T89988 CGY45E 71519054 IC50 = 400 nM T89988 C29BZD 71519055 IC50 = 290 nM T89988 CR1IO9 71519224 IC50 = 34 nM T89988 CQ8F3O 71519225 IC50 = 1800 nM T89988 CE07SH 71519226 IC50 = 16 nM T89988 C2FE7Q 71519227 IC50 = 95 nM T89988 CP25YK 71519381 IC50 = 61 nM T89988 C3CT1R 71530223 IC50 = 22 nM T89988 C7XGD2 71552097 IC50 = 36 nM T89988 CQ31YB 71552260 IC50 = 39 nM T89988 CO3WL9 71552261 IC50 = 50 nM T89988 CU2R7W 71576618 Ki = 2.3 nM T89988 CI0GU8 71660496 IC50 > 48500 nM T89988 C5GE1T 71716742 IC50 = 88 nM T89988 CI8Q1K 71717723 Ki = 0.6 nM T89988 CP5NQ2 71718331 Ki = 1 nM T89988 CZ5C6V 71718930 Ki = 2 nM T89988 CC8JQ9 71719547 Ki = 1 nM T89988 CG30CF 71719764 IC50 = 130 nM T89988 CC80KL 71768688 IC50 = 16 nM T89988 CPX2W4 71768689 IC50 = 8.7 nM T89988 C4KUV6 71768721 IC50 = 62 nM T89988 CX39OE 71768722 IC50 = 2 nM T89988 CE5BJ7 71768725 IC50 = 16 nM T89988 C9NHU5 71768755 IC50 = 4 nM T89988 C65HBS 71768794 IC50 = 14 nM T89988 COE81F 71768798 IC50 = 59 nM T89988 C9ZKP0 71768830 IC50 = 29 nM T89988 CN9TQ3 71768831 IC50 = 330 nM T89988 CHQ15U 71768862 IC50 = 340 nM T89988 C8ERI3 71768864 IC50 = 27 nM T89988 C7ZY1J 71768865 IC50 = 1.5 nM T89988 C54JLD 71768897 IC50 = 370 nM T89988 CV53CZ 71768899 IC50 = 2130 nM T89988 CJY2C5 71768900 IC50 = 6.6 nM T89988 CKU6V5 71768931 IC50 = 35 nM T89988 C4EM1B 72945827 IC50 = 950 nM T89988 C1G5DP 72945830 IC50 = 69 nM T89988 C8RLE2 72946008 IC50 = 41 nM T89988 CDG6A2 72946010 IC50 = 99 nM T89988 C3N7RS 72946013 IC50 = 39 nM T89988 C37UZP 72946198 IC50 = 31 nM T89988 CF65HX 72946199 IC50 = 65 nM T89988 CI8Z0Q 72946200 IC50 = 82 nM T89988 C9FLS6 72946202 IC50 = 629 nM T89988 CA4L5S 72946204 IC50 = 126 nM T89988 CPA9G7 72946205 IC50 = 180 nM T89988 CF7WR3 72946381 IC50 = 28 nM T89988 CX82VR 72946384 IC50 = 1300 nM T89988 C7X2ZL 72946387 IC50 = 29 nM T89988 C16RLM 72946775 IC50 = 45 nM T89988 CP21YZ 72946982 IC50 = 118 nM T89988 CB51JH 72947191 IC50 = 87 nM T89988 CZR9S4 72947193 IC50 = 21 nM T89988 CMB52G 72947411 IC50 = 33 nM T89988 CN8U7J 72947413 IC50 = 395 nM T89988 CU9NB5 72947593 IC50 = 770 nM T89988 C7TIG1 72947595 IC50 = 27 nM T89988 CJQ04K 72948000 IC50 = 57 nM T89988 CO42FH 72948001 IC50 = 71 nM T89988 CFC70R 72948004 IC50 = 68 nM T89988 CXR6G5 73334813 Ki = 2.4 nM T89988 CT1RD0 73351183 EC50 = 630 nM T89988 CX9B4F 76167595 Ki = 2 nM T89988 CT2QF9 76314234 IC50 = 81 nM T89988 CSFB37 76314242 IC50 = 62 nM T89988 C2TLD8 76315270 IC50 = 10 nM T89988 CQT3F1 76321527 IC50 = 152 nM T89988 C8N9QM 76325121 IC50 = 1215 nM T89988 C1XL3H 76333441 IC50 = 39 nM T89988 C3Y0WL 76335990 IC50 = 300 nM T89988 CW1AZ2 86642531 IC50 = 0.13 nM T89988 C7TRY9 89844945 IC50 = 2.2 nM T89988 CE2Z4C 89845025 IC50 = 1.2 nM T89988 CTP94N 89845031 IC50 = 5 nM T89988 CN3DO5 89853102 IC50 = 1280 nM T89988 C9PSW7 90656015 IC50 = 5700 nM T89988 CTU8Z7 90656016 IC50 > 20000 nM T89988 C6N5DH 90656017 IC50 = 3170 nM T89988 CYTC65 90656018 IC50 > 20000 nM T89988 CZ1S2O 90656019 IC50 = 16100 nM T89988 C15QNG 90656020 IC50 = 2200 nM T89988 C3CAQ0 90656021 IC50 = 81 nM T89988 C6OI3C 90656022 IC50 = 180 nM T89988 C4FI1L 90656023 IC50 > 20000 nM T89988 CW4Z3B 90656024 IC50 > 20000 nM T89988 CK6QN4 90656025 IC50 = 30 nM T89988 CO73FL 90656026 IC50 = 190 nM T89988 COW7U5 90656027 IC50 = 0.25 nM T89988 C6ENV5 100951623 EC50 > 10000 nM T89988 CU29LP 118723021 Ki = 74 nM T89988 CZ1PV5 118723406 Ki = 270 nM T89988 CUGV43 118723408 Ki = 66 nM T89988 CK3S2X 118723411 Ki = 139 nM T89988 CP24GA 118723412 Ki = 90 nM T89988 CP10RK 118734571 Ki = 15 nM T89988 C2BWS4 118734572 Ki = 2.2 nM T89988 C75BLE 118734573 Ki = 31 nM T89988 CCP2L0 118734574 Ki = 4.6 nM T89988 C20SEZ 118734575 Ki = 15 nM T89988 CSOP75 118734576 Ki = 21 nM T89988 C8ZK9S 118734577 Ki = 4.9 nM T89988 CYOI62 118734578 Ki = 1.6 nM T89988 C94AOU 118734579 Ki = 4.4 nM T89988 CR8IY6 118734580 Ki = 13 nM T89988 C52KYS 118734581 Ki = 23 nM T89988 C5U1JI 118734582 Ki = 13 nM T89988 CDRN42 118734583 Ki = 7.9 nM T89988 C82WOS 118734584 Ki = 1.2 nM T89988 C50DNS 118734671 Ki = 49 nM T89988 CW7J0V 118734675 Ki = 55 nM T89988 CQ9N3Y 118734676 Ki = 11 nM T89988 CRJL05 118734678 Ki = 39 nM T89988 C52TGP 118734679 Ki = 75 nM T89988 C7RI8B 118734680 Ki = 10 nM T89988 CRF84D 118734681 Ki = 41 nM T89988 CGV9X0 118734682 Ki = 10 nM T89988 CAQ14V 118734683 Ki = 23 nM T89988 C47KNY 118734684 Ki = 12 nM T89988 CW08JS 118734685 Ki = 3.4 nM T89988 CIE93O 118734686 Ki = 2 nM T89988 C5K1DJ 118734687 Ki = 4.5 nM T89988 CNB69H 118734688 Ki = 13 nM T89988 CM9AJ8 118734689 Ki = 83 nM T89988 C1LNT2 118734690 Ki = 24 nM T89988 CG8FH2 118734691 Ki = 2 nM T89988 CT3MG4 118734692 Ki = 4.6 nM T89988 CRXS03 118734693 Ki = 199 nM T89988 CHPC27 118734694 Ki = 137 nM T89988 CA81LN 122178127 IC50 = 62 nM T89988 C2AWE9 122178128 IC50 = 1.8 nM T89988 CXN3E7 122181144 IC50 = 684 nM T89988 CQY5H1 122181145 IC50 = 7540 nM T89988 CJB1F7 122181146 IC50 = 1240 nM T89988 CM9PW3 122181147 IC50 = 180 nM T89988 C0V1MG 122181148 IC50 = 12000 nM T89988 C20HIU 122181149 IC50 = 318 nM T89988 CA0QB2 122181150 IC50 = 89 nM T89988 C1VM5E 122181151 IC50 = 462 nM T89988 CGRW01 122181152 IC50 = 163 nM T89988 C5KA8W 122181153 IC50 = 173 nM T89988 CYA7Z5 122181235 IC50 = 1600 nM T89988 CE5WF4 122181236 IC50 = 353 nM T89988 C8DC5N 122181237 IC50 = 6100 nM T89988 C0X6MH 122181238 IC50 = 17 nM T89988 CMOW05 127025086 IC50 = 1.2 nM T89988 CQD1C7 127025087 IC50 < 0.45 nM T89988 C2Y6EC 127025088 IC50 = 1.1 nM T89988 CGT84Q 127025089 IC50 = 9.2 nM T89988 CG32CV 127025091 IC50 = 41 nM T89988 CPU3B6 127025092 IC50 = 7.4 nM T89988 C5WC3V 127025093 IC50 = 1.7 nM T89988 CR5H4I 127025159 IC50 = 5406 nM T89988 CFL76Q 127025160 IC50 = 6605 nM T89988 CVJS82 127025444 IC50 = 9737 nM T89988 CZ80IQ 127025445 IC50 = 928 nM T89988 C7PY8T 127025446 IC50 = 284 nM T89988 CCWU81 127025447 IC50 = 254 nM T89988 C6BX2Y 127025448 IC50 = 1685 nM T89988 C1CE3P 127025460 IC50 = 150 nM T89988 C5AY2X 127025461 IC50 = 210 nM T89988 CWAU40 127025462 IC50 = 6151 nM T89988 C6XA7T 127025728 IC50 = 2637 nM T89988 CMXT79 127025729 IC50 = 3700 nM T89988 C57XLF 127025730 IC50 = 328 nM T89988 CHYK14 127026243 IC50 = 2.3 nM T89988 CL04JF 127027624 IC50 = 301 nM T89988 C8RK9W 127027625 IC50 = 744 nM T89988 CPUA26 127027626 IC50 = 3480 nM T89988 CL0DQ7 127027627 IC50 > 10000 nM T89988 C17CTI 127027628 IC50 = 114 nM T89988 CE45ZO 127027955 IC50 = 69 nM T89988 C1RSE3 127027956 IC50 = 249 nM T89988 C6SP7M 127028586 IC50 = 700 nM T89988 C71UIE 127028587 IC50 = 3418 nM T89988 C0ML7J 127028588 IC50 = 2967 nM T89988 C3YF7I 127028589 IC50 > 10000 nM T89988 CMJA67 127028590 IC50 = 1600 nM T89988 CU7DL4 127028591 IC50 = 8200 nM T89988 C7QWB2 127028592 IC50 = 438 nM T89988 CQ10RI 127029034 IC50 = 2.7 nM T89988 CPKQ90 127036603 IC50 = 550 nM T89988 CA4I9H 127036934 IC50 = 3700 nM T89988 CSD1X5 132572938 IC50 = 140 nM T89988 CK8XQ2 135981707 IC50 = 170 nM T89988 C9YAI3 136030597 IC50 > 10000 nM T89988 C2WT5B 137654404 IC50 = 3000 nM T89988 CGRA79 145953092 IC50 = 2502 nM T89988 C7ZFD4 145953762 IC50 = 638 nM T89988 CWVF94 145953765 IC50 = 3864 nM T89988 CQ2J5K 145954490 IC50 = 74 nM T89988 C0RE7W 145954949 IC50 = 336 nM T89988 C4BWN2 145955877 IC50 = 4936 nM T89988 CX96RN 145960485 IC50 = 720 nM T89988 C4R1XZ 145960924 IC50 = 7833 nM T89988 CW4N2T 145961260 IC50 = 1566 nM T89988 CB02GJ 145961667 IC50 = 19390 nM T89988 CKO9D2 145961759 IC50 = 1614 nM T89988 CD3IV4 145961961 IC50 = 1821 nM T89988 C32SJE 145961982 IC50 = 61 nM T89988 C4GL7Y 145962429 IC50 = 1261 nM T89988 CG3FT6 145962546 IC50 = 1731 nM T89988 C7Y8BD 145962575 IC50 = 390 nM T89988 C40AEX 145962604 IC50 = 5053 nM T89988 CNZ32U 145962608 IC50 = 550 nM T89988 CABC91 145962732 IC50 = 2466 nM T89988 CV8F3U 145963369 IC50 = 195 nM T89988 C72LVY 145963552 IC50 = 12330 nM T89988 C3UR2C 145963612 IC50 = 4450 nM T89988 CXR41S 145963669 IC50 = 2971 nM T89988 CFN4J8 145996522 Ki = 1.549 nM T89988 CXT09R 154572822 IC50 = 0.4 nM T89988 COP6C1 155491018 Ki = 0.3802 nM T89988 CVQ31N 155513284 Ki = 1.549 nM T89988 CW6CH0 155513605 Ki = 22.39 nM T89988 C7R1SZ 155513751 Ki = 316 nM T89988 CM7Y9H 155514261 IC50 = 8709.64 nM T89988 C70IOJ 155518928 Ki = 15.49 nM T89988 CMJU07 155520385 Ki = 4.074 nM T89988 CZ29FQ 155521447 Ki = 15 nM T89988 CN61LU 155522058 Ki = 51.29 nM T89988 CKX47L 155522874 Ki = 173.78 nM T89988 CBKQ30 155523645 Ki = 14.45 nM T89988 CW0R6Z 155526680 Ki = 213.8 nM T89988 CKR1O4 155527193 Ki = 20.89 nM T89988 C86OHR 155529593 IC50 = 1.9 nM T89988 CZ7TU0 155529754 Ki = 5.495 nM T89988 CCOP08 155530253 Ki = 154.88 nM T89988 CVS37C 155531379 IC50 = 1.4 nM T89988 C52QOY 155531561 Ki = 6.31 nM T89988 C0GAF2 155534565 Ki = 5.37 nM T89988 CF6DQ7 155535265 Ki = 158.49 nM T89988 CL0O2E 155535293 Ki = 3.467 nM T89988 CFDV10 155536512 Ki = 104.6 nM T89988 CE5SU4 155539148 Ki = 102.33 nM T89988 CK4I2Z 155540563 Ki = 288.4 nM T89988 CZ04TG 155540798 Ki = 2.188 nM T89988 CT9V0L 155541801 Ki = 2.951 nM T89988 CW71FQ 155543260 Ki = 3.467 nM T89988 C7FS8U 155545321 Ki = 12.88 nM T89988 C4J1ZL 155545804 Ki = 154.88 nM T89988 CRKZ36 155550777 Ki = 21.88 nM T89988 C03TXA 155551912 Ki = 2.089 nM T89988 CU32YB 155553131 Ki = 22.91 nM T89988 CYW9U3 155553573 Ki = 7.2 nM T89988 C3DB6L 155553917 Ki = 1.8 nM T89988 CT4NC3 155554106 Ki = 0.8318 nM T89988 C80LBZ 155554273 Ki = 0.6 nM T89988 C7X6VW 155559153 Ki = 66 nM T89988 C0TCG8 155560784 Ki = 2.455 nM T89988 C06NGD 155562719 Ki = 0.871 nM T89988 CF8JW6 155563012 Ki = 1.445 nM T89988 D0RM7J 44353447 IC50 = 17 nM T53904 D01SPD 69669724 IC50 = 480 nM T53904 D09NCT 53392492 IC50 = 54000 nM T53904 CMO39B 7493 Ki > 300000 nM T53904 CR85KY 10253 IC50 > 1000000 nM T53904 C5H7QS 9837038 IC50 = 91090 nM T53904 CUP73E 10103626 IC50 = 1000000 nM T53904 CM6Q3H 11788622 IC50 > 1000000 nM T53904 C4XC1Z 13548097 IC50 > 1000000 nM T53904 CYRZ62 15662041 IC50 = 24000 nM T53904 CCAM68 22959876 IC50 > 100000 nM T53904 C30EMN 24701909 IC50 = 18370 nM T53904 CZ8WG7 24831508 IC50 = 3.5 nM T53904 CUMF70 46899605 IC50 > 100000 nM T53904 C2DBN5 46899607 IC50 > 100000 nM T53904 C3G4QK 46899609 IC50 > 100000 nM T53904 CLK96Z 46899763 IC50 > 100000 nM T53904 CBOM64 46899765 IC50 > 100000 nM T53904 CA56RL 49831102 IC50 = 1.8 nM T53904 CU63QR 49847377 IC50 = 0.2 nM T53904 CZT4I8 49847378 IC50 = 0.3 nM T53904 CA72PE 49847379 IC50 = 1.1 nM T53904 CJ7H2B 49847753 IC50 = 1.4 nM T53904 C4V7EW 49848258 IC50 = 1.2 nM T53904 CP8TS6 49848895 IC50 = 0.3 nM T53904 C9COF5 49848896 IC50 = 0.3 nM T53904 CK0B1G 49848897 IC50 = 0.2 nM T53904 CP61VJ 49849002 IC50 = 0.3 nM T53904 C42SBF 49849005 IC50 = 1.4 nM T53904 CBM62Z 49849007 IC50 = 0.4 nM T53904 C05SEW 49849008 IC50 = 0.2 nM T53904 C78SAD 49849115 IC50 = 2.1 nM T53904 CF64IJ 49849120 IC50 = 0.2 nM T53904 CC9EB4 49849122 IC50 = 0.4 nM T53904 C2ORV5 49849123 IC50 = 6 nM T53904 CU7O4S 52942802 IC50 = 500000 nM T53904 C28RDF 54746913 IC50 = 3.6 nM T53904 C35JDV 54746961 IC50 = 3.6 nM T53904 CDL06K 54746964 IC50 = 2.4 nM T53904 C34DJP 57384236 IC50 = 0.8 nM T53904 CEOC15 57384237 IC50 = 2.1 nM T53904 CY50WC 57384238 IC50 = 2.3 nM T53904 C7S0ZR 57384239 IC50 = 1.8 nM T53904 C2XN1G 57384481 IC50 = 1.1 nM T53904 CR73IZ 57384482 IC50 = 0.7 nM T53904 CR2M5H 57384483 IC50 = 0.3 nM T53904 CQ72HI 57384749 IC50 = 3.7 nM T53904 C68KGE 57384750 IC50 = 1.6 nM T53904 CVK29R 57386523 IC50 = 1.7 nM T53904 C9S8MU 57386524 IC50 = 1.4 nM T53904 CMC8H6 57386782 IC50 = 1.1 nM T53904 CCT5D4 57386783 IC50 = 0.2 nM T53904 CC30XZ 57386784 IC50 = 8.2 nM T53904 C79BXP 57386785 IC50 = 0.9 nM T53904 CM6DV7 57387028 IC50 = 1.2 nM T53904 C0GS4F 57387282 IC50 = 0.3 nM T53904 C0TL9C 57387283 IC50 = 0.8 nM T53904 CRV2P5 57387539 IC50 = 0.2 nM T53904 CAU3G9 57387540 IC50 = 0.3 nM T53904 CL2AO8 57387541 IC50 = 0.3 nM T53904 C0XWL8 57387542 IC50 = 0.4 nM T53904 CC4DK0 57387775 IC50 = 1 nM T53904 C8DB9I 57387776 IC50 = 1 nM T53904 C73OLG 59186234 IC50 = 240 nM T53904 CCB65L 59603622 IC50 = 480 nM T53904 C4VU7J 70688210 IC50 = 5.5 nM T53904 CO7H3Q 71133989 IC50 = 2.1 nM T53904 C7K3JM 89812866 IC50 = 240 nM T53904 CUX19J 117632648 IC50 = 30000 nM T53904 CSEB74 117705981 IC50 = 570 nM T53904 CI5X2G 118978277 IC50 = 6.8 nM T53904 CH7WL3 118978299 IC50 = 11 nM T53904 CB3I9Z 118978325 IC50 = 6.3 nM T53904 CWH4I0 118978339 IC50 = 14 nM T53904 C6XD3H 118978341 IC50 = 3.3 nM T53904 CDBK07 118981498 IC50 = 2.2 nM T53904 CB23LS 118981525 IC50 = 12 nM T53904 C9F6RL 118981536 IC50 = 6.2 nM T53904 CF1E6T 118981546 IC50 = 11 nM T53904 C1ABC5 118981554 IC50 = 3.7 nM T53904 CR05OQ 118981555 IC50 = 5 nM T53904 CE9U5L 118981600 IC50 = 2.4 nM T53904 CO5XH7 118981638 IC50 = 4.9 nM T53904 CV84HB 118981731 IC50 = 3.1 nM T53904 CW89CV 118982285 IC50 = 3.8 nM T53904 C51RST 121245332 IC50 = 3.2 nM T53904 C2LI6C 121245745 IC50 = 5.9 nM T53904 C27WIY 121246694 IC50 = 27 nM T53904 C71YRT 121246805 IC50 = 2.3 nM T53904 CJU6X7 121246821 IC50 = 1.4 nM T53904 C1X3HT 121246837 IC50 = 4.9 nM T53904 C2UY6K 121246848 IC50 = 2.1 nM T53904 CRO04U 122540293 IC50 = 280 nM T53904 CQ5R9P 122540295 IC50 = 57 nM T53904 CB9K4N 122540308 IC50 = 34 nM T53904 C5ZIL1 122540317 IC50 = 67 nM T53904 C1KS9O 122540318 IC50 = 770 nM T53904 CPN71M 122540325 IC50 = 90 nM T53904 C5BFA8 122540341 IC50 = 1800 nM T53904 CPZ8I3 122540362 IC50 = 140 nM T53904 C6IEP4 122540388 IC50 = 50 nM T53904 CJ0RB3 122540392 IC50 = 39 nM T53904 CTG8N2 122540437 IC50 = 140 nM T53904 C6S2RC 122540446 IC50 = 13 nM T53904 CO34NP 122540461 IC50 = 1280 nM T53904 CZ0OW9 122540496 IC50 = 220 nM T53904 C6XL8K 122540512 IC50 = 3900 nM T53904 C81EIY 122540553 IC50 = 1370 nM T53904 C1ZMX3 122540617 IC50 = 10 nM T53904 C2EFG9 122540625 IC50 = 670 nM T53904 CK81UQ 122540630 IC50 = 8 nM T53904 C8K1DC 122540636 IC50 = 84 nM T53904 CTCL51 122540637 IC50 = 170 nM T53904 CD3VP5 122540661 IC50 = 6100 nM T53904 CI2ZX4 122540667 IC50 = 1870 nM T53904 CZ8M5Q 122540675 IC50 = 550 nM T53904 C3DOK6 122540683 IC50 = 74 nM T53904 CM1X0A 122540685 IC50 = 830 nM T53904 CLV75P 122540689 IC50 = 52 nM T53904 C38VFM 122540702 IC50 = 140 nM T53904 CAIU61 122540718 IC50 = 460 nM T53904 C1QXU7 122540722 IC50 = 25 nM T53904 C2LK0Y 122540724 IC50 = 34 nM T53904 CS61XJ 122540744 IC50 = 200 nM T53904 CYC48U 122540745 IC50 = 160 nM T53904 C1VOT7 122540750 IC50 = 460 nM T53904 CLT3K0 122540759 IC50 = 70 nM T53904 CG9T1H 134328388 IC50 = 270 nM T53904 CT57ZH 136069450 IC50 = 0.2 nM T53904 CFT9R3 136069453 IC50 = 0.5 nM T53904 CRPQ42 136069494 IC50 = 1.3 nM T53904 CK8Z3V 136069521 IC50 = 1.9 nM T53904 CPY1B2 136069522 IC50 = 17 nM T53904 CX0OM4 136069523 IC50 = 11 nM T53904 C6EU4D 136069524 IC50 = 38 nM T53904 CQA2Z1 136069531 IC50 = 4.5 nM T53904 CCH31A 136069532 IC50 = 0.4 nM T53904 CH8GV7 136069561 IC50 = 5.6 nM T53904 CQ1FS4 136069563 IC50 = 2 nM T53904 CQTB32 136205798 IC50 = 1.1 nM T53904 CV8QP3 136205832 IC50 = 0.2 nM T53904 CB93EM 136205833 IC50 = 0.5 nM T53904 C23FVD 137633446 IC50 > 100000 nM T53904 CPU1L2 137636406 IC50 = 5600 nM T53904 C8TN4G 137636671 IC50 = 55000 nM T53904 CG3F4E 137637795 IC50 > 100000 nM T53904 C1M6HB 137638932 IC50 = 2500 nM T53904 CFB79N 137641310 IC50 = 80000 nM T53904 C0DTF7 137641650 IC50 > 10000 nM T53904 C6PRQ9 137641829 IC50 > 10000 nM T53904 C34MZN 137642369 IC50 > 100000 nM T53904 CC7JI6 137646003 IC50 = 24000 nM T53904 C8NLW2 137648088 IC50 = 48000 nM T53904 CGX30Y 137648213 IC50 = 26000 nM T53904 CEWP67 137648313 IC50 > 10000 nM T53904 C78LJT 137649345 IC50 > 10000 nM T53904 CJ76HR 137649729 IC50 > 10000 nM T53904 C9AJ4B 137652165 IC50 > 10000 nM T53904 CU2IS6 137653429 IC50 = 9600 nM T53904 C25TUJ 137653793 IC50 > 10000 nM T53904 CD8HL9 137655479 IC50 > 10000 nM T53904 CWG40Z 137655745 IC50 > 10000 nM T53904 C9C3RJ 137657820 IC50 = 1300 nM T53904 C5DV0L 137658554 IC50 > 10000 nM T53904 C4XQH5 137659524 IC50 = 18000 nM T53904 CVB05O 137660951 IC50 = 28000 nM T53904 CD7LE9 137661677 IC50 = 61000 nM T53904 C2TB0E 137662021 IC50 = 26000 nM T53904 CG7R3L 155559901 IC50 = 3.2 nM T53904 D07IOY 10365 IC50 = 1500 nM T53904 D08IZY 3080614 IC50 = 842 nM T58449 D03ZBT 11626560 IC50 > 10000 nM T58449 D05SBO 46220502 IC50 = 300 nM T58449 D00UZR 5330286 IC50 > 10000 nM T58449 D05ADP 160355 IC50 = 480 nM T58449 D0CY1B 6420138 Ki > 10000 nM T58449 D0LF1U 5287969 IC50 = 875 nM T58449 D0S5RC 3025986 IC50 = 62 nM T58449 CB9F1O 447961 Ki = 70 nM T58449 C6A3LY 447962 Ki = 4012 nM T58449 CVX20F 9842276 IC50 = 1300 nM T58449 CVE1W8 10024433 Ki = 2804 nM T58449 C1KX3P 10248401 Ki > 10000 nM T58449 C9J3RM 10320107 Ki = 1080 nM T58449 CMY9D2 10340715 Ki > 10000 nM T58449 CC3L8Z 10430000 Ki > 10000 nM T58449 C69HPR 11257553 Ki = 2.3 nM T58449 CIWA03 11632150 Ki = 243 nM T58449 CEV5X2 11646645 Ki = 171 nM T58449 C2CVI7 11647020 Ki = 1395 nM T58449 C93KHF 11718021 Ki = 370 nM T58449 CJSV21 11744184 Ki > 10000 nM T58449 CCX39H 15979015 IC50 = 11000 nM T58449 CBV7T6 15979138 IC50 = 1000 nM T58449 CI5Q2D 15979261 IC50 = 410 nM T58449 C3ZC4Y 15979393 IC50 = 480 nM T58449 C6Z4CR 15979397 IC50 > 10000 nM T58449 C4D5UF 15979518 IC50 = 260 nM T58449 C1JMA7 15979519 IC50 > 2000 nM T58449 CARL15 15979630 IC50 > 3700 nM T58449 CXYU20 15979633 IC50 > 10000 nM T58449 CQD02P 15979747 IC50 > 10000 nM T58449 C8MGY5 15979751 IC50 = 210 nM T58449 CF9SK3 15979868 IC50 = 170 nM T58449 C7UEG5 15980106 IC50 = 160 nM T58449 CPJY86 15980107 IC50 = 705 nM T58449 CU87FW 15980108 IC50 > 10000 nM T58449 CQH37B 15980109 IC50 = 340 nM T58449 CB7JU8 15980233 IC50 > 10000 nM T58449 C7BS2R 16037674 IC50 > 10000 nM T58449 CB2H4D 16037675 IC50 = 530 nM T58449 C42DYS 16091079 IC50 > 20000 nM T58449 C5VPH9 16129448 IC50 = 2730 nM T58449 CQHK69 23646624 IC50 = 1500 nM T58449 C7YG1N 24759534 IC50 = 30 nM T58449 C4EG8R 24993189 IC50 > 10000 nM T58449 C5HZF2 44413509 IC50 = 20 nM T58449 C3D4FG 44413527 IC50 = 190 nM T58449 C3VRO9 44557921 IC50 > 10000 nM T58449 CGO1J5 46830766 Ki = 4240 nM T58449 CF7HK2 46830767 Ki = 2556 nM T58449 C2HJ1X 46830768 Ki = 2149 nM T58449 CKL1V8 49798556 IC50 > 20000 nM T58449 CCL3R5 49867929 IC50 = 21 nM T58449 C1DV2B 56932125 IC50 = 1760 nM T58449 C2VK6A 57404485 IC50 = 2100 nM T58449 CK6T1C 57404486 IC50 = 350 nM T58449 CQ80BX 57404487 IC50 = 317 nM T58449 CR1B9I 57867443 IC50 > 10000 nM T58449 C42IGJ 57867446 IC50 = 910 nM T58449 C18QUW 57867482 IC50 = 870 nM T58449 CIZ91X 57867490 IC50 = 960 nM T58449 C1VFJ8 57867505 IC50 = 940 nM T58449 C3Z5KS 57867516 IC50 > 10000 nM T58449 CFB7Q4 57867522 IC50 > 10000 nM T58449 CXJ63M 59603829 IC50 = 53 nM T58449 CQEU96 59603842 IC50 = 4.1 nM T58449 C37NKO 67129970 IC50 > 10000 nM T58449 CK80LJ 67130050 IC50 > 10000 nM T58449 C7GRV2 68755406 IC50 > 10000 nM T58449 CM8LY4 70681104 IC50 > 10000 nM T58449 CHC4P3 70685325 IC50 > 10000 nM T58449 C49QWD 70691636 IC50 = 26 nM T58449 CBE67N 71731769 IC50 < 5 nM T58449 CYG95S 72707651 IC50 = 1876 nM T58449 CNP0V5 72707724 IC50 = 1788 nM T58449 CU4A5Q 72707728 IC50 = 1645 nM T58449 CZAM98 72707790 IC50 = 1642 nM T58449 CP13FK 72707853 IC50 = 1423 nM T58449 C7VA5U 78161839 IC50 = 0.13 nM T58449 C2Y1RF 78162193 IC50 < 5 nM T58449 C4NM0V 78162195 IC50 < 5 nM T58449 CWR57U 78357763 IC50 = 27 nM T58449 C1HW4B 89735655 IC50 < 10 nM T58449 C8W9KV 91844733 IC50 = 40 nM T58449 CQCX41 118737057 IC50 > 10000 nM T58449 C4WGC7 119081415 IC50 = 194 nM T58449 C2BEH5 121443990 IC50 > 100 nM T58449 CP4Q7B 121444083 IC50 = 20 nM T58449 C9MIL3 122188249 IC50 = 841 nM T58449 C53AYQ 122188250 IC50 > 10000 nM T58449 CZO41H 122188251 IC50 > 10000 nM T58449 CLW25J 122188252 IC50 = 9244 nM T58449 C23PIE 122188253 IC50 > 10000 nM T58449 CE41KZ 122188254 IC50 > 10000 nM T58449 CHQT85 122188255 IC50 > 10000 nM T58449 CLAD59 122188256 IC50 > 10000 nM T58449 C3BXR2 122188258 IC50 > 10000 nM T58449 C67GYV 122188259 IC50 > 10000 nM T58449 CG8VX5 122188261 IC50 > 10000 nM T58449 C9ZKA1 122188262 IC50 > 10000 nM T58449 CQF9I2 122188263 IC50 > 10000 nM T58449 COGF57 122188264 IC50 > 10000 nM T58449 CPQ89G 122188266 IC50 = 3590 nM T58449 CVEB28 122188271 IC50 = 8750 nM T58449 C5E7WK 122188272 IC50 > 10000 nM T58449 CWIR28 122188273 IC50 > 10000 nM T58449 CB6I5A 122188274 IC50 > 10000 nM T58449 CA8VH1 122188275 IC50 = 1811 nM T58449 C2D5TF 122188281 IC50 > 10000 nM T58449 C93VST 122188282 IC50 = 1680 nM T58449 C4X7SD 122192466 IC50 > 10000 nM T58449 CM0A3E 124134260 IC50 < 100 nM T58449 COF75Z 126970673 IC50 = 300 nM T58449 C1SP3H 127030849 IC50 = 2780 nM T58449 CDJQ32 127051599 IC50 = 21 nM T58449 C1MTG5 134543905 IC50 = 20 nM T58449 C37ITY 135414445 IC50 = 6500 nM T58449 C5AG7L 135414460 IC50 = 56 nM T58449 CLXB05 135438541 IC50 = 300 nM T58449 CR48OH 135468068 IC50 = 39 nM T58449 CPE67T 135487516 IC50 = 11 nM T58449 CJ4V0A 135508121 IC50 = 310 nM T58449 C2JA3F 135520167 IC50 = 180 nM T58449 C25MKU 135559056 IC50 = 1300 nM T58449 CHW54V 135559057 IC50 = 4900 nM T58449 C4CJG9 135559058 IC50 > 100000 nM T58449 CCQ4J8 135559059 IC50 = 25 nM T58449 CDN21F 135559061 IC50 = 34 nM T58449 C8BJV6 135559062 IC50 = 18 nM T58449 CS4HA0 135559063 IC50 = 4000 nM T58449 C2BHG0 135559064 IC50 = 57 nM T58449 CMF9Y8 135559065 IC50 = 420 nM T58449 C61XZP 135559066 IC50 = 2300 nM T58449 CPC03V 135559067 IC50 = 480 nM T58449 C8G2TS 135559068 IC50 = 7000 nM T58449 CI1E8V 137634241 IC50 > 10000 nM T58449 CVU63L 139582016 IC50 = 3100 nM T58449 C8PH9S 139582017 IC50 = 17000 nM T58449 CR2GW6 145994117 IC50 = 3600 nM T58449 CYHW79 155530843 IC50 = 20 nM T58449 C1IHY8 155533514 IC50 > 200 nM T58449 C8OC5N 155537111 IC50 < 20 nM T58449 CETH36 155557337 IC50 < 20 nM T58449 CLXN40 155565350 IC50 = 193 nM T58449 D00ERW 44444843 Ki > 1525 nM T58449 D01MNK 25125014 IC50 = 250 nM T58449 D02QAZ 11612883 IC50 = 197 nM T58449 D03DZO 11715767 IC50 > 10000 nM T58449 D0LO5B 73602827 IC50 = 3.2 nM T58449 D0YZ7H 9797370 IC50 = 56700 nM T15139 CD74LR 292706 Ki = 27000 nM T15139 CGA5F2 346675 IC50 = 57500 nM T15139 CTHK18 895402 IC50 = 5600 nM T15139 C3M0VW 1838078 IC50 > 100000 nM T15139 C2GL0X 1869842 IC50 < 50000 nM T15139 CDT51Y 1951286 IC50 < 50000 nM T15139 C9N5XB 2026662 IC50 > 100000 nM T15139 CGX7T5 2120805 IC50 > 100000 nM T15139 CO9Y3Z 4355463 IC50 = 6800 nM T15139 CXS9F6 4566836 IC50 = 5400 nM T15139 CKZ7V6 4674993 IC50 = 7000 nM T15139 C9ID6V 4912070 IC50 > 100000 nM T15139 C1O3RJ 5010967 IC50 = 37200 nM T15139 CV8FZ1 6875399 IC50 = 35700 nM T15139 C1KF4O 8615611 IC50 > 57000 nM T15139 CFX96S 15544085 IC50 = 6600 nM T15139 CMV5X1 17011425 IC50 > 100000 nM T15139 CBXC05 24424330 IC50 = 8700 nM T15139 CF9J3R 49852772 IC50 = 37000 nM T15139 C9QSP2 49852889 IC50 = 8900 nM T15139 C4HU6B 49852897 IC50 = 11000 nM T15139 CYZC96 49852943 IC50 = 6400 nM T15139 C7AEH1 49853067 IC50 = 14000 nM T15139 C47SDM 49853091 IC50 = 10000 nM T15139 CES9G3 49853100 IC50 = 13000 nM T15139 C78HFB 49853142 IC50 = 37000 nM T15139 CU21EH 49853203 IC50 > 57000 nM T15139 C64EUF 49853209 IC50 = 6300 nM T15139 C2ZN7D 49853294 IC50 = 5300 nM T15139 C6ZCA3 49853368 EC50 = 17500 nM T15139 CYIC61 53257121 IC50 = 21000 nM T15139 CKA74G 101879233 IC50 = 68900 nM T15139 CMLW04 102205482 IC50 = 22800 nM T15139 C6W2ZN 118796328 EC50 = 2300 nM T15139 CMO57H 118947294 IC50 < 50000 nM T15139 C0X8KJ 118947349 IC50 > 100000 nM T15139 CBOS58 118947388 IC50 > 100000 nM T15139 CU53JP 118947412 IC50 < 50000 nM T15139 C1XZF7 118947462 IC50 > 100000 nM T15139 CB39WZ 118947481 IC50 > 100000 nM T15139 C8RCS4 118947495 IC50 > 100000 nM T15139 CN5J3Z 118947501 IC50 = 50000 nM T15139 CIZ72P 118947502 IC50 < 50000 nM T15139 CB4W1C 118947563 IC50 < 50000 nM T15139 C5MH7P 118947571 IC50 < 50000 nM T15139 C3PJB8 121485232 IC50 = 50000 nM T15139 C7BJ6G 121485242 IC50 = 10000 nM T15139 C91HSG 121485258 IC50 = 21000 nM T15139 CFIH36 121485269 IC50 = 8700 nM T15139 CEDA24 122418186 IC50 = 33000 nM T15139 C26VJM 130407999 IC50 = 30 nM T15139 C7P5EJ 130408291 IC50 = 10 nM T15139 CY65ND 130418263 IC50 = 153 nM T15139 CV1U2H 130429937 IC50 = 88100 nM T15139 CQ6AI9 130429939 IC50 = 160700 nM T15139 C6SFT7 130429940 IC50 = 9300 nM T15139 CR27LM 130429942 IC50 > 200000 nM T15139 CD5F7E 130429947 IC50 > 200000 nM T15139 C0MVF4 130429950 IC50 > 100000 nM T15139 CT48EP 130429983 IC50 > 200000 nM T15139 CHB9F5 130429986 IC50 > 100000 nM T15139 C18LPS 130429999 IC50 > 200000 nM T15139 C94VCX 130430007 IC50 > 200000 nM T15139 CNGD28 130430011 IC50 > 200000 nM T15139 C8LUX7 130430025 IC50 > 200000 nM T15139 CUE3P2 134429273 IC50 = 31000 nM T15139 CQAO64 134429274 IC50 = 8300 nM T15139 CW06KT 134429275 IC50 = 5800 nM T15139 CO2P5Y 134429276 IC50 = 9900 nM T15139 C5AD7I 134429279 IC50 = 12000 nM T15139 C5DS8E 134437716 IC50 = 19000 nM T15139 C8MWK9 134437740 IC50 = 5700 nM T15139 CW0DZ5 134437744 IC50 = 6300 nM T15139 C5NDX1 134437746 IC50 = 41000 nM T15139 C8T6YN 134437750 IC50 = 22000 nM T15139 CD8B6U 134437753 IC50 = 30000 nM T15139 CEL49B 134437755 IC50 = 20000 nM T15139 CPT52N 134437756 IC50 = 20000 nM T15139 C3OYN0 134437757 IC50 = 17000 nM T15139 C2OT5L 134437812 IC50 = 26000 nM T15139 CO8Q3N 134437824 IC50 = 15000 nM T15139 CH90ED 134437828 IC50 = 40000 nM T15139 C3ML0D 134437829 IC50 = 39000 nM T15139 CMS49R 134437832 IC50 = 38000 nM T15139 CXI18Q 134437838 IC50 = 9200 nM T15139 C3GPI7 134437841 IC50 = 11000 nM T15139 CMX8P1 134437848 IC50 = 11000 nM T15139 C8SW4G 134437869 IC50 = 6500 nM T15139 C8NKX2 134437870 IC50 = 11000 nM T15139 CCV31P 134437872 IC50 = 10000 nM T15139 CPNO39 134437877 IC50 = 7200 nM T15139 CVM23J 134437914 IC50 = 7700 nM T15139 CZQB64 134437925 IC50 = 17000 nM T15139 CY4AV9 135403154 IC50 = 34800 nM T15139 CTK6F0 136937731 IC50 > 100000 nM T15139 CBX7R0 137522167 IC50 = 1400 nM T15139 CR5O3C 137647070 IC50 > 100000 nM T15139 C3GKP5 137651355 IC50 > 100000 nM T15139 CS3QB9 137655343 IC50 > 100000 nM T15139 C21INE 137657956 IC50 > 100000 nM T15139 CG5HS1 138753630 Ki = 214 nM T15139 CVM80R 138756828 IC50 = 100 nM T15139 C8QC5T 138756829 IC50 = 400 nM T15139 CPR5Y3 138756830 IC50 = 300 nM T15139 CG3L7H 138756831 IC50 = 3 nM T15139 CV3D1R 138911337 IC50 = 2000 nM T15139 C21PYB 142427688 IC50 = 8 nM T15139 CZC62Y 142427749 IC50 = 4 nM T15139 CU4T6V 145960504 IC50 = 8000 nM T15139 CHX5N9 145960596 IC50 = 9700 nM T15139 CT9XH5 145960621 IC50 = 21000 nM T15139 CI40NB 145960758 IC50 = 4300 nM T15139 C7RW0X 145960898 IC50 = 23000 nM T15139 CU1IK7 145961091 IC50 = 50000 nM T15139 CNY09E 145961156 IC50 = 15000 nM T15139 C3P8LH 145961174 IC50 = 16000 nM T15139 CHQ56V 145961472 IC50 = 7300 nM T15139 C0T6SZ 145961708 IC50 = 59000 nM T15139 CP4LA9 145962107 IC50 = 24000 nM T15139 CAC5D9 145962456 IC50 = 14000 nM T15139 CY2KN7 145962789 IC50 = 8700 nM T15139 C3U9VD 145963193 IC50 = 12000 nM T15139 CS49BK 145963368 IC50 = 16000 nM T15139 CM64FH 145963685 IC50 = 7300 nM T15139 C96DLG 155510912 IC50 = 2500 nM T15139 C7VUG8 155512349 IC50 = 72 nM T15139 CSCH29 155513145 IC50 = 14 nM T15139 C32NXU 155515150 IC50 = 3300 nM T15139 CZ19YB 155516063 IC50 = 1580 nM T15139 CDK81A 155516285 IC50 = 15 nM T15139 CL2W0D 155516426 IC50 = 5200 nM T15139 CE2P4T 155516866 IC50 = 53800 nM T15139 CIAJ65 155516908 IC50 = 81 nM T15139 CWCT76 155517908 IC50 > 100000 nM T15139 CCN07T 155517974 IC50 = 287 nM T15139 CB2HW7 155518094 IC50 = 100 nM T15139 CZJ72G 155518421 IC50 = 6700 nM T15139 CK15XH 155518761 IC50 = 2368 nM T15139 CRH20E 155519110 IC50 > 100000 nM T15139 C24BQW 155522173 IC50 = 23200 nM T15139 C1NH8X 155523199 IC50 = 34 nM T15139 C73NSI 155525342 IC50 = 37 nM T15139 CY90TS 155525802 IC50 = 58 nM T15139 C2XIY9 155526005 IC50 = 39600 nM T15139 C7Q1EB 155526382 IC50 = 33000 nM T15139 C72UBT 155526686 IC50 = 25 nM T15139 CMGW68 155526835 IC50 = 22000 nM T15139 CM02HQ 155527973 IC50 = 1294 nM T15139 C0AUE1 155528104 IC50 = 2300 nM T15139 CB92UN 155529283 IC50 = 23400 nM T15139 CA58ZG 155531601 IC50 = 235 nM T15139 C17OHV 155532142 IC50 = 38100 nM T15139 CION96 155534368 IC50 = 30 nM T15139 CN12SJ 155535053 IC50 = 12100 nM T15139 CJN2M3 155536090 IC50 = 301 nM T15139 CB6D3O 155536637 IC50 > 100000 nM T15139 CT7L3S 155536748 IC50 = 1330 nM T15139 C6ND9J 155536777 IC50 = 5200 nM T15139 C4KTE5 155537075 IC50 = 51 nM T15139 C6LEK7 155537339 IC50 = 5700 nM T15139 CT5YL8 155537379 IC50 > 100000 nM T15139 CLB65J 155537992 IC50 > 100000 nM T15139 CTP4L0 155538389 IC50 = 900 nM T15139 C5GP6H 155538643 IC50 = 25 nM T15139 CS38OJ 155538775 IC50 = 1300 nM T15139 CKGW41 155541540 IC50 = 55400 nM T15139 CUT17I 155542117 IC50 = 4300 nM T15139 CT42PF 155542308 IC50 = 824 nM T15139 CXQ9T4 155542332 IC50 = 1400 nM T15139 C94XQG 155542973 IC50 = 28 nM T15139 C4D5ZQ 155544502 IC50 = 3100 nM T15139 C0OTJ1 155544677 IC50 = 209000 nM T15139 C1M4ZS 155545662 IC50 = 439 nM T15139 C86AEZ 155546222 IC50 > 100000 nM T15139 C3DON9 155546449 IC50 = 16200 nM T15139 CDM02P 155547534 IC50 = 42100 nM T15139 C2YUJ1 155550274 IC50 = 11700 nM T15139 CM8WK4 155550368 IC50 > 100000 nM T15139 C47GNZ 155552547 IC50 = 22000 nM T15139 C42UCY 155553773 IC50 = 235 nM T15139 CX16DK 155554240 IC50 = 70 nM T15139 C49EHO 155555646 IC50 = 12200 nM T15139 CNI86P 155556782 IC50 = 990 nM T15139 CWLB78 155557800 IC50 = 33700 nM T15139 CF03HW 155558291 IC50 = 341 nM T15139 CEIJ65 155558670 IC50 > 100000 nM T15139 C20MVN 155559066 IC50 = 1950 nM T15139 CMQP04 155559154 IC50 = 800 nM T15139 CD60PE 155559613 IC50 = 5830 nM T15139 CF4LH0 155562166 IC50 = 6000 nM T15139 C27QFZ 155562355 IC50 = 370 nM T15139 C3MN6X 155563952 IC50 = 21500 nM T15139 C5BP6R 155567916 IC50 = 100000 nM T15139 COJ5M8 155569162 IC50 = 1460 nM T15139 CU8K5P 155569553 IC50 = 28 nM T26368 D06ZII 969472 Ki > 15000 nM T26368 D07JVL 3016 Ki = 15 nM T26368 D0L9GG 2118 EC50 = 10 nM T26368 D0T1WN 5732 EC50 > 3000 nM T26368 D02XYB 3058746 IC50 = 4.6 nM T26368 D0CH7C 57336276 Ki = 4.7 nM T26368 D0HO2T 23581869 Ki = 230 nM T26368 D0Z9HW 23630026 Ki = 1680 nM T26368 C1W5EF 114888 Ki = 0.85 nM T26368 C7SZ9E 613843 IC50 > 10000 nM T26368 C12NWX 2729103 IC50 > 10000 nM T26368 CO61AF 2820320 IC50 > 10000 nM T26368 C59BWK 2820473 IC50 > 10000 nM T26368 CCX58U 9865233 Ki = 1.1 nM T26368 C7BA0Z 9908880 Ki = 2.3 nM T26368 CPC3U1 9971547 Ki = 6 nM T26368 CUSM85 10221761 Ki = 33.3 nM T26368 C15NXT 10926766 EC50 = 650 nM T26368 CK1S7J 10927005 EC50 = 375 nM T26368 CWK02D 10936672 EC50 = 94 nM T26368 C09PCZ 10971225 EC50 = 323 nM T26368 CJB1V2 11035207 EC50 = 291 nM T26368 CBV36I 11047145 EC50 = 231 nM T26368 CWO70Q 11673720 Ki = 2 nM T26368 CL4XD0 11783674 EC50 = 74 nM T26368 CTI32Y 15680235 EC50 = 1000 nM T26368 CZK75V 44364548 EC50 = 439 nM T26368 C0FN6W 44364725 EC50 = 112 nM T26368 CE8F3Y 44364734 EC50 = 90 nM T26368 COH5G6 44364735 EC50 = 111 nM T26368 C2VHW7 44364747 EC50 = 491 nM T26368 CZL2P0 44364907 EC50 = 38 nM T26368 CCX08E 44364918 EC50 = 346 nM T26368 C6J0GP 44561356 IC50 = 210 nM T26368 C9UW4V 44561357 IC50 = 550 nM T26368 CZR6A5 44561358 IC50 > 10000 nM T26368 C4IF7B 44561386 IC50 = 1000 nM T26368 C0PC5E 44561389 Ki = 83 nM T26368 CP5WT1 44561431 Ki = 500 nM T26368 CPJC74 44561432 Ki = 0.65 nM T26368 C0L1FI 44561433 Ki = 9.8 nM T26368 C4S7HF 44561434 Ki = 2610 nM T26368 CB4I1E 44561435 Ki = 166 nM T26368 C6J7DH 44561436 Ki > 300 nM T26368 CO2QA8 44561437 Ki = 182 nM T26368 CDN1A9 44561475 Ki = 369 nM T26368 CN24OF 46229639 Ki = 2364 nM T26368 C1BZN5 71584335 Ki = 24.9 nM T26368 CQ91VU 118278442 Ki = 7.9 nM T26368 CH0D4J 130439777 Ki = 55 nM T26368 C56XBU 130439778 Ki = 5000 nM T26368 C9N8LW 130439889 Ki = 79 nM T26368 C89LNZ 136118605 IC50 = 201 nM T26368 D06SOQ 6918451 Ki = 0.66 nM T26368 D09IHE 6918583 Ki = 1.4 nM T26368 D0E7PY 11624499 Ki = 4.6 nM T26368 D0M4CP 5081 Ki = 3.1 nM T26368 D0O9MG 5311203 Ki = 0.45 nM T25956 D02YNI 9936746 IC50 > 33000 nM T25956 D07SDQ 969516 IC50 = 6500 nM T25956 D0M2TS 71600087 IC50 = 63 nM T25956 D0PH9I 118693659 Ki < 10000 nM T25956 D0U2BH 65064 IC50 = 30000 nM T25956 CM2RK5 67254 IC50 = 118500 nM T25956 CK5QD7 73588 IC50 = 4850 nM T25956 CQ8A5W 91330 IC50 = 13700 nM T25956 CX16AI 122042 IC50 = 260 nM T25956 CHU6D4 343829 IC50 = 106000 nM T25956 CXCB27 393166 IC50 = 2430 nM T25956 CHR5Q8 395862 IC50 = 8280 nM T25956 CH1DM6 769739 IC50 = 6200 nM T25956 CO8HA9 832572 IC50 = 2600 nM T25956 COJ29X 890649 IC50 = 11000 nM T25956 CGZ7Y8 900269 IC50 = 14000 nM T25956 CM2Z5Q 1285941 Ki = 400 nM T25956 CS96HU 1367211 IC50 = 1800 nM T25956 CG1I7T 1550234 IC50 = 111000 nM T25956 CJWR09 1561807 IC50 = 81000 nM T25956 CS05BM 1600566 IC50 = 244100 nM T25956 C4EZ0H 1652812 IC50 = 660 nM T25956 C5DXU9 1797299 IC50 = 700 nM T25956 C6XQA3 1797300 IC50 = 700 nM T25956 CBIP78 2133789 IC50 = 1100 nM T25956 C8E9HY 2221149 IC50 = 1980 nM T25956 CBK1D6 2295854 IC50 = 2200 nM T25956 C4T8OV 2325816 IC50 = 8030 nM T25956 C1YZ8I 2327942 IC50 = 9350 nM T25956 CTVG84 2328663 IC50 = 8140 nM T25956 COTE61 2408437 IC50 = 24700 nM T25956 C1LNM0 2467794 IC50 = 12900 nM T25956 CZE13I 2816786 IC50 = 6740 nM T25956 C5F2BD 2854538 IC50 = 150000 nM T25956 CQUY78 2871948 Ki = 400 nM T25956 CAY86S 3312427 IC50 = 6200 nM T25956 C54MWY 3493274 IC50 = 1100 nM T25956 CG8F2A 3683950 IC50 = 15200 nM T25956 CMK3Q0 3801109 IC50 = 2800 nM T25956 CWJ93L 5124087 IC50 = 3700 nM T25956 C13OPQ 5352088 IC50 = 7000 nM T25956 C4FKS8 5467476 IC50 = 233000 nM T25956 CG1LV3 7333990 IC50 > 50000 nM T25956 CK4GM7 7574135 IC50 = 3000 nM T25956 CSX8V7 7897116 IC50 = 510 nM T25956 C2FM4R 9875131 IC50 = 5000 nM T25956 CH41UK 9992116 IC50 = 5350 nM T25956 C7NT2X 10311918 IC50 = 275000 nM T25956 CUD8X4 10355367 IC50 = 5710 nM T25956 C2QTW8 11052198 IC50 = 23000 nM T25956 C6EMN5 11114773 IC50 = 5000 nM T25956 CCTY51 11135781 Ki = 3900 nM T25956 C8OCA4 12005893 IC50 = 1800 nM T25956 CXP5S8 12006282 IC50 = 2000 nM T25956 C7U9KW 13099766 IC50 = 5740 nM T25956 C29QHR 13374635 IC50 = 1100 nM T25956 CP82EX 14117443 IC50 = 1900 nM T25956 C1ZIE7 16203604 IC50 = 168000 nM T25956 CW6TU0 16203606 IC50 = 5000 nM T25956 C1DM9I 18783165 IC50 = 95000 nM T25956 CWS8N7 22121498 IC50 = 1100 nM T25956 CI0FB7 24320099 IC50 = 1000 nM T25956 C46RLS 42609873 IC50 = 3000 nM T25956 C6Q7IJ 44564009 IC50 = 28000 nM T25956 CO3UF4 44564514 IC50 = 9900 nM T25956 CRK2E6 44564516 IC50 = 14400 nM T25956 C52BJH 44571034 IC50 = 3.2 nM T25956 C6BQ2N 44580829 Ki = 5100 nM T25956 CU46TX 45032907 IC50 = 7500 nM T25956 C87QKN 50899265 IC50 = 70 nM T25956 CG3PR6 52912222 IC50 = 31622.78 nM T25956 C4XCJ0 53257845 IC50 = 5920 nM T25956 CBOE48 56669892 IC50 = 5320 nM T25956 C6I7VX 60201924 IC50 < 5000 nM T25956 C1X7DC 60201925 IC50 < 5000 nM T25956 C6YD5U 60201926 IC50 = 5000 nM T25956 CLGW91 60201927 IC50 < 5000 nM T25956 CI3MA8 60201928 IC50 < 5000 nM T25956 C5OPX2 60201929 IC50 < 5000 nM T25956 CPR3T5 60201930 IC50 = 5000 nM T25956 C8EDT9 60202083 IC50 < 5000 nM T25956 CJTM92 60202084 IC50 < 5000 nM T25956 CCX28H 60202085 IC50 = 5000 nM T25956 CZ47SK 60202086 IC50 = 5000 nM T25956 C2Q0NP 60202087 IC50 < 5000 nM T25956 CD84NS 71481176 IC50 = 11 nM T25956 CBX37Z 72201043 IC50 = 58000 nM T25956 CX9CV2 76853637 IC50 = 57500 nM T25956 CQ1V6U 86302322 IC50 = 9190 nM T25956 CS3W6O 90667751 IC50 = 61900 nM T25956 CZBD29 90667752 IC50 = 151900 nM T25956 CF4W8Q 90667754 IC50 = 95300 nM T25956 CTA46H 91826273 Ki = 2000 nM T25956 CM9Y5S 102127780 IC50 = 3300 nM T25956 C8ZVB6 118734156 IC50 = 9800 nM T25956 CB58PX 118735300 IC50 = 2100 nM T25956 C6J0QZ 118735301 IC50 = 1600 nM T25956 CM29SP 118735302 IC50 = 5900 nM T25956 CIKU37 118735303 IC50 = 1500 nM T25956 C2CQ5J 118735304 IC50 = 11400 nM T25956 CPH4W9 118735305 IC50 = 8000 nM T25956 C96FHE 118735307 IC50 = 8500 nM T25956 CYWS40 118735308 IC50 = 5400 nM T25956 CA8P3R 118735309 IC50 = 31400 nM T25956 C0UR4G 118735310 IC50 = 4200 nM T25956 C6NI1C 118735317 IC50 = 26400 nM T25956 C3TG2V 118735320 IC50 = 1600 nM T25956 C0QY8M 118958122 IC50 = 60 nM T25956 CUWX94 119081692 IC50 = 270 nM T25956 CB83MK 121271792 IC50 = 51 nM T25956 CDH8M4 121373418 IC50 = 1.3 nM T25956 C47QXT 121376807 IC50 = 30 nM T25956 C7PRX6 124351359 IC50 = 750 nM T25956 CC1AX6 125920038 IC50 = 45000 nM T25956 C8C1ZL 126458860 IC50 = 3400 nM T25956 CD3AJ2 126797002 IC50 = 3700 nM T25956 CV4D8T 127030247 IC50 = 7000 nM T25956 CLB9N0 127033602 IC50 = 5000 nM T25956 CPIG89 127033885 IC50 = 22 nM T25956 CU2O8R 127045845 IC50 = 14100 nM T25956 CGDN94 132275066 IC50 = 1.2 nM T25956 CY46VZ 135423665 IC50 = 3100 nM T25956 C4KDT9 135457159 IC50 > 50000 nM T25956 CPY8E7 139341516 IC50 = 4000 nM T25956 C3HJI2 139341518 IC50 = 26900 nM T25956 CWK82L 139341520 IC50 > 33000 nM T25956 C3DGA7 139341522 IC50 = 17800 nM T25956 C4CHN3 139341523 IC50 = 34700 nM T25956 CRW7P5 139341524 IC50 = 5400 nM T25956 C98TAG 139341527 IC50 = 25100 nM T25956 CJ01EC 139341528 IC50 = 25100 nM T25956 C5F7OS 139341530 IC50 = 15600 nM T25956 COY2D4 139341532 IC50 = 57000 nM T25956 C6BV5E 139341541 IC50 = 16500 nM T25956 CWM81B 139341544 IC50 = 18600 nM T25956 CF1VL4 139341553 IC50 > 33000 nM T25956 CF8LU1 139341570 IC50 > 5000 nM T25956 C3SVA5 139341572 IC50 = 2200 nM T25956 CL9XU2 139341575 IC50 > 33000 nM T25956 C69JHS 139341584 IC50 > 33000 nM T25956 C7IN1U 139341589 IC50 > 100000 nM T25956 C0HT4J 139341591 IC50 > 100000 nM T25956 CF2D6W 139341726 IC50 > 100000 nM T25956 CI1H2T 139341727 IC50 > 100000 nM T25956 C9K8YX 139341747 IC50 > 100000 nM T25956 C4YMW6 139341818 IC50 > 100000 nM T25956 C8ZQ2U 141736359 IC50 = 1780 nM T25956 C5VNM4 141736367 IC50 = 49 nM T25956 C3YGJ5 145948689 IC50 = 200000 nM T25956 C96NCH 145950955 IC50 = 4450 nM T25956 C3ZV1O 145952497 IC50 = 5550 nM T25956 CB7R2C 145952522 IC50 = 8800 nM T25956 CTE74G 145954441 IC50 = 2510 nM T25956 C5WX1Y 145954899 IC50 = 52000 nM T25956 CRHG03 145955376 IC50 > 10000 nM T25956 CKO51W 145955422 IC50 > 10000 nM T25956 C3D8LO 145955588 IC50 = 60000 nM T25956 CN5YO3 145957310 IC50 = 510 nM T25956 C8JI5E 145957556 IC50 = 250000 nM T25956 C7C5WL 145958595 IC50 = 970 nM T25956 CM19OV 145959971 IC50 > 10000 nM T25956 C2OG9K 145964185 IC50 = 3900 nM T25956 C2I9YJ 145969602 IC50 = 3900 nM T25956 C15GYL 145973549 IC50 = 3900 nM T25956 CAD6O9 145975385 IC50 = 3900 nM T25956 CNHR01 145987968 IC50 > 50000 nM T25956 CBRE71 146047136 IC50 = 3857 nM T25956 CI1F6L 146204973 IC50 > 1000 nM T25956 CXG1V9 146204995 IC50 = 10 nM T25956 C2AJO8 146205056 IC50 = 2.6 nM T25956 CQM7N8 146205057 IC50 = 3 nM T25956 C9HWQ8 146205061 IC50 = 4 nM T25956 CH8E2N 146205066 IC50 = 1.9 nM T25956 CO4S3M 146205067 IC50 = 10 nM T25956 C1N5IH 146205070 IC50 = 7.5 nM T25956 CZN7D5 146205179 IC50 = 4.3 nM T25956 CZLO67 146205182 IC50 = 46 nM T25956 C5TXC2 146205184 IC50 = 3.7 nM T25956 CZU3B7 146205188 IC50 > 1000 nM T25956 CL4T3H 146205226 IC50 = 4.2 nM T25956 CUA52Y 146205228 IC50 = 2.4 nM T25956 CJ7Y0W 146205434 IC50 = 2.4 nM T25956 CY7GI4 146205498 IC50 = 30 nM T25956 CGYR94 146205502 IC50 = 14 nM T25956 CR3P4I 146205515 IC50 = 10 nM T25956 C8Z9OM 146205579 IC50 = 1.8 nM T25956 CQ1IX3 151484729 IC50 = 9610 nM T25956 CLZ34P 155512196 IC50 > 1000 nM T25956 CVJT64 155512236 IC50 = 290 nM T25956 C2WJ4O 155513273 IC50 > 10000 nM T25956 CYUW30 155514843 IC50 = 1600 nM T25956 CCI7T9 155515172 IC50 > 10000 nM T25956 C7E1TC 155516066 IC50 = 7310 nM T25956 CKM42V 155516765 IC50 > 10000 nM T25956 C2DI1Q 155516796 IC50 = 1130 nM T25956 CKR7F9 155518500 IC50 > 500 nM T25956 CG95RD 155519099 IC50 = 22 nM T25956 C2A1YU 155519665 IC50 = 2000 nM T25956 C5J8XK 155519829 IC50 = 470 nM T25956 CHD7V8 155520793 IC50 = 230 nM T25956 CMW49Z 155521226 IC50 = 860 nM T25956 C1MZC7 155522494 IC50 > 10000 nM T25956 CNL8O1 155522829 IC50 = 560 nM T25956 CE35PR 155523264 IC50 = 200 nM T25956 C3Y5XO 155523600 IC50 = 5000 nM T25956 C1SLG3 155524393 IC50 = 2400 nM T25956 CIA61E 155524527 IC50 = 5000 nM T25956 C63TIU 155524913 IC50 < 10000 nM T25956 CZ2FD5 155525448 IC50 = 6050 nM T25956 C87AZN 155525893 IC50 < 10000 nM T25956 C9OP3H 155527488 IC50 = 7130 nM T25956 C2T3OR 155528202 IC50 = 1800 nM T25956 C4XW9I 155528393 IC50 = 6000 nM T25956 CHR4K5 155528532 IC50 = 160 nM T25956 CKUM79 155528818 IC50 = 8600 nM T25956 C3LEV4 155529291 IC50 = 1800 nM T25956 CQEF61 155531348 IC50 > 10000 nM T25956 C8YNB3 155531682 IC50 < 10000 nM T25956 CHW29R 155532177 IC50 = 1950 nM T25956 C32MLY 155532996 IC50 > 10000 nM T25956 C1RPU0 155533512 IC50 > 2000 nM T25956 CK9S7N 155534073 IC50 > 10000 nM T25956 CBL5O0 155534637 IC50 > 10000 nM T25956 C9WB4Q 155534723 IC50 = 7400 nM T25956 C2RP4X 155535364 IC50 = 4400 nM T25956 C3W8XH 155536530 IC50 = 4 nM T25956 C95OQP 155536635 IC50 = 620 nM T25956 C1FEC3 155537172 IC50 = 580 nM T25956 CS3F4K 155537389 IC50 = 1.1 nM T25956 CFBE34 155538503 IC50 = 11 nM T25956 CX2Y9E 155538946 IC50 > 10000 nM T25956 CP4TW3 155539039 IC50 = 1700 nM T25956 C5KX7C 155539735 IC50 = 1530 nM T25956 CB5XE8 155539809 IC50 = 190 nM T25956 CZDW67 155540096 IC50 > 10000 nM T25956 C9KTW6 155540252 IC50 = 9800 nM T25956 CDR92H 155540348 IC50 = 5400 nM T25956 C7EOQ9 155540603 IC50 = 5000 nM T25956 C96MUR 155540976 IC50 = 3000 nM T25956 CIAT68 155542185 IC50 > 10000 nM T25956 CS3FY1 155543664 IC50 > 10000 nM T25956 CV0F2H 155544116 IC50 = 670 nM T25956 C9SUY7 155544858 IC50 = 1.3 nM T25956 COC7P0 155546490 IC50 = 2200 nM T25956 CTE76J 155547116 IC50 = 4600 nM T25956 CV56PN 155547836 IC50 = 4060 nM T25956 COHT62 155547999 IC50 = 8600 nM T25956 CX3UR0 155548318 IC50 = 2070 nM T25956 C71RPH 155548492 IC50 < 10000 nM T25956 C84GSF 155549456 IC50 < 10000 nM T25956 CP6AN5 155554496 IC50 > 10000 nM T25956 CUQ5F8 155556860 IC50 > 10000 nM T25956 CR0Y5U 155558481 IC50 = 24000 nM T25956 C8PUJ7 155558550 IC50 = 3730 nM T25956 CVL3T0 155559427 IC50 > 10000 nM T25956 CMD2A9 155559553 IC50 = 1400 nM T25956 C1TPW8 155559730 IC50 = 1800 nM T25956 CT3P5J 155559844 IC50 = 1170 nM T25956 CCY7V1 155559876 IC50 = 2800 nM T25956 CA9RW0 155560578 IC50 > 10000 nM T25956 C65CMJ 155561106 IC50 > 100 nM T25956 CQ70NE 155561894 IC50 = 73 nM T25956 CKR5A2 155563315 IC50 = 420 nM T25956 C8FD7C 155563587 IC50 = 1600 nM T25956 C2MNY1 155564022 IC50 > 10000 nM T25956 C1H9VW 155564054 IC50 > 10000 nM T25956 C2VR1B 155564237 IC50 > 10000 nM T25956 CT8S7I 155564925 IC50 = 4800 nM T25956 CK25GR 155565190 IC50 = 10000 nM T25956 C68CBM 155565352 IC50 = 12600 nM T25956 CM3SV1 155565651 IC50 = 7400 nM T25956 CY9GF7 155566211 IC50 = 12 nM T25956 CUK53M 155566805 IC50 > 10000 nM T25956 CP3B8C 155566822 IC50 = 7000 nM T25956 CZ5U4A 155568100 IC50 = 5800 nM T25956 CUDW40 155568215 IC50 = 1800 nM T25956 C4DE3Y 155568219 IC50 > 10000 nM T25956 D03XXT 72201027 IC50 = 230 nM T25956 D05RDP 992586 IC50 = 330 nM T25956 D07MTM 403 IC50 > 500000 nM T25956 D08XXD 17815 IC50 = 1400 nM T25956 D0E6JS 167551 IC50 = 8500 nM T25956 D0M6YZ 25226432 IC50 = 5000 nM T25956 D0P0IE 10205 IC50 = 2000 nM T25956 D0W3NA 87642 IC50 = 45940 nM T25956 D0YL8Z 1285940 IC50 = 9.8 nM T63414 D01BYB 5957 EC50 = 780000 nM T63414 D07QTG 66553218 IC50 = 5.012 nM T63414 D0CS2C 10161381 IC50 = 10 nM T63414 D0F4JK 11547499 IC50 = 1.3 nM T63414 D0H2UB 5361 EC50 = 92000 nM T63414 D0VI4N 90409366 IC50 = 3.467 nM T63414 D00PVH 16679492 IC50 = 39.81 nM T63414 D0FR8L 73442861 IC50 = 0.33 nM T63414 D0F8DL 176155 IC50 = 5000 nM T63414 CI15DO 265893 IC50 = 22.4 nM T63414 C1WDR8 331254 IC50 = 281.84 nM T63414 CX9F0T 331256 IC50 = 109.65 nM T63414 CCKT54 344276 IC50 = 414 nM T63414 CA3W5F 707096 IC50 = 522 nM T63414 CIWV85 746996 IC50 > 100000 nM T63414 CMUV80 766793 IC50 = 69800 nM T63414 CEBX03 779113 IC50 > 100000 nM T63414 CGJ9S2 921624 IC50 = 40800 nM T63414 C7BL5H 1478602 IC50 = 478 nM T63414 CN5T0V 1485975 IC50 = 125.89 nM T63414 CYV85L 2320735 IC50 > 10000 nM T63414 C3NPH7 2741121 IC50 = 501.19 nM T63414 CPD81K 2811018 IC50 = 320 nM T63414 CO8D1M 2812882 IC50 = 1400 nM T63414 C0S6BO 2831480 IC50 = 100 nM T63414 CR3FI4 2926477 IC50 = 4540 nM T63414 C6NAF0 2933256 IC50 = 7.943 nM T63414 C5J6IN 2941710 IC50 = 3981.07 nM T63414 C5HD9G 3079322 IC50 > 1000 nM T63414 C1RN5V 3454885 IC50 = 398.11 nM T63414 C47QZJ 3709284 IC50 = 398.11 nM T63414 CA5I3R 3872625 IC50 > 10000 nM T63414 CY68AQ 3932023 IC50 = 600 nM T63414 C81JUQ 4023622 IC50 = 3981.07 nM T63414 CM7W9S 4423333 IC50 = 125.89 nM T63414 C1V6ZX 4563797 IC50 = 501.19 nM T63414 C69OFV 4768671 IC50 = 4240 nM T63414 CPA28C 5052387 IC50 = 600 nM T63414 CJQ6M9 5151658 IC50 = 158.49 nM T63414 CN25AH 5176829 IC50 > 10000 nM T63414 CW1Q3Z 5229632 IC50 = 398.11 nM T63414 C01FHC 6466568 IC50 = 4960 nM T63414 C2WRS6 8923923 IC50 = 64.57 nM T63414 CL6DZ9 9045905 IC50 = 158.49 nM T63414 CT1K8I 9209741 IC50 = 1000 nM T63414 CSH1M6 9268807 IC50 = 79.43 nM T63414 CZDJ08 9270241 IC50 > 1000 nM T63414 CO1KY9 9821690 IC50 < 10000 nM T63414 CXE7T9 9821948 IC50 = 7.943 nM T63414 CU30FS 9878599 IC50 = 15848.93 nM T63414 CS05ET 9896790 IC50 = 1.3 nM T63414 CVL25E 9926842 IC50 = 10 nM T63414 CM74RK 9948588 IC50 = 158.49 nM T63414 CH05KP 9985155 IC50 = 50.12 nM T63414 C5VI1R 10086144 IC50 = 71.2 nM T63414 CST2B3 10115466 IC50 = 63.1 nM T63414 C05QVB 10117302 IC50 = 350 nM T63414 CYO93C 10126799 IC50 = 300 nM T63414 CM9OX5 10129577 IC50 = 132 nM T63414 C5JMC4 10139090 IC50 < 10000 nM T63414 CXYD23 10139173 IC50 < 10000 nM T63414 CT3SL2 10150143 IC50 = 4 nM T63414 COQU26 10153625 IC50 = 18.5 nM T63414 C2F5QT 10153639 IC50 = 97.7 nM T63414 CWHT56 10153662 IC50 = 100 nM T63414 CL30XQ 10153683 IC50 = 380 nM T63414 CVBZ07 10153700 IC50 = 12.3 nM T63414 CV71DN 10161380 IC50 = 0.23 nM T63414 CCA84W 10175779 IC50 = 70.8 nM T63414 C9RKJ2 10181729 IC50 < 10000 nM T63414 CMLT35 10190472 IC50 = 6 nM T63414 C0TJ1A 10197227 IC50 = 19.95 nM T63414 CKDG89 10202422 IC50 = 79.43 nM T63414 C0FK5C 10204578 IC50 = 63.1 nM T63414 CF7J5N 10212541 IC50 = 5.8 nM T63414 CZ29UQ 10219050 IC50 = 84.1 nM T63414 CDA5R8 10219058 IC50 = 15.8 nM T63414 C84RHX 10225191 IC50 < 10000 nM T63414 CBF8K0 10238746 IC50 = 15.85 nM T63414 CYJP45 10240451 IC50 = 101 nM T63414 C6ARI8 10240476 IC50 = 1122 nM T63414 C9IC5W 10276962 IC50 < 10000 nM T63414 C61FKR 10279659 IC50 = 500 nM T63414 C1GDY4 10290336 IC50 = 170 nM T63414 CXO1K8 10290342 IC50 = 79.43 nM T63414 CF6CX0 10290368 IC50 = 15.1 nM T63414 C5UX9N 10290391 IC50 = 600 nM T63414 C9DV4H 10290419 IC50 = 5.8 nM T63414 C0CY3U 10290496 IC50 = 176 nM T63414 C31FWT 10295970 IC50 < 10000 nM T63414 CSHM81 10297818 IC50 < 10000 nM T63414 CW28SB 10310632 IC50 = 10 nM T63414 C7Z0QM 10312629 IC50 = 28.8 nM T63414 C76XQR 10312667 IC50 = 13.5 nM T63414 C1C9ZI 10312693 IC50 = 12.59 nM T63414 CX56LQ 10312737 IC50 = 31.1 nM T63414 CF9JG2 10312739 IC50 = 33.9 nM T63414 CLN6Z9 10546931 IC50 = 560 nM T63414 COK26H 11007110 IC50 = 65.3 nM T63414 CPO5B9 11115244 IC50 < 1000 nM T63414 C2DJ7W 11167023 IC50 = 63.1 nM T63414 CCBW78 11179231 IC50 = 50.12 nM T63414 CJ3W8P 11187581 IC50 = 3 nM T63414 CRK5N7 11189340 IC50 = 63.1 nM T63414 CC21XM 11190463 IC50 = 50.12 nM T63414 C4V9WN 11199715 IC50 = 930 nM T63414 CK7I8C 11209712 IC50 = 630.96 nM T63414 C1Y5LT 11212938 IC50 = 100 nM T63414 CRS95A 11213305 IC50 = 100 nM T63414 CK61OS 11223687 IC50 = 31.62 nM T63414 CQM28B 11225321 IC50 = 100 nM T63414 COS8U3 11225680 IC50 = 31.62 nM T63414 CQ0C9T 11231942 IC50 = 316.23 nM T63414 CTWN36 11259677 IC50 = 79.43 nM T63414 CDOR07 11269479 IC50 = 100 nM T63414 CFPO95 11270845 IC50 = 10 nM T63414 C2XZ5B 11279679 IC50 = 10 nM T63414 CP25KE 11281239 IC50 = 63.1 nM T63414 CS6GY2 11294314 IC50 = 630.96 nM T63414 CA3I2Y 11327640 IC50 = 50.12 nM T63414 CIT65D 11350742 IC50 = 31.62 nM T63414 C8Z9LM 11351050 IC50 = 79.43 nM T63414 C4NPA1 11351142 IC50 = 39.81 nM T63414 C2XVW3 11351651 IC50 = 10 nM T63414 C6OE5H 11352109 IC50 = 50.12 nM T63414 C20GWS 11361743 IC50 = 79.43 nM T63414 CNE40H 11373994 IC50 = 63.1 nM T63414 CBI5L3 11374948 IC50 = 79.43 nM T63414 CI3RZ0 11386290 IC50 = 3.162 nM T63414 C8GJW2 11414871 IC50 = 125.89 nM T63414 CZF7H4 11418470 IC50 = 63.1 nM T63414 C2BE5J 11419335 IC50 <= 199.53 nM T63414 C07IEJ 11441307 IC50 = 25.12 nM T63414 C9S7LP 11442400 IC50 = 501.19 nM T63414 CRBG65 11453381 IC50 = 50.12 nM T63414 CBD6P3 11464418 IC50 = 19.95 nM T63414 CEXZ01 11465129 IC50 = 63.1 nM T63414 CQJ05C 11486676 IC50 = 63.1 nM T63414 C59BYU 11500704 IC50 = 31.62 nM T63414 CM2XS3 11503827 IC50 = 63.1 nM T63414 C92MUN 11507787 IC50 = 501.19 nM T63414 CWX01V 11508020 IC50 = 14.45 nM T63414 C2ND7T 11508207 IC50 = 3981.07 nM T63414 CAGV64 11509663 IC50 = 28.18 nM T63414 CBJ89G 11515022 IC50 = 39.81 nM T63414 CN9IS7 11516301 IC50 = 125.89 nM T63414 CR0MX4 11523472 IC50 = 23.99 nM T63414 C07CTD 11530196 IC50 = 12.59 nM T63414 CQG79J 11530593 IC50 = 25.12 nM T63414 CP3DM2 11530961 IC50 = 109.65 nM T63414 CZ40XE 11531460 IC50 = 63.1 nM T63414 CAW1T2 11537311 IC50 = 20.89 nM T63414 C1S2XY 11537418 IC50 = 199.53 nM T63414 CY52PW 11540045 IC50 = 100 nM T63414 C1RL5A 11543793 IC50 = 25118.86 nM T63414 C08CHM 11544727 IC50 = 18.2 nM T63414 C5A3FH 11546350 IC50 = 158.49 nM T63414 C9MZT6 11564932 IC50 = 25118.86 nM T63414 CIJ24Y 11566345 IC50 = 794.33 nM T63414 CTN61H 11573809 IC50 = 19.95 nM T63414 CXM10I 11574070 IC50 = 12.59 nM T63414 CNW65B 11602877 IC50 = 12589.25 nM T63414 C49UPR 11609203 IC50 = 15848.93 nM T63414 CC8NB2 11610500 IC50 = 12.59 nM T63414 C2QDJ4 11616778 IC50 = 63.1 nM T63414 C5JN4R 11625340 IC50 = 15 nM T63414 CV4I8J 11630893 IC50 = 100 nM T63414 C5T6EI 11639163 IC50 = 54.95 nM T63414 C57ZHK 11644745 IC50 = 7943.28 nM T63414 COVY38 11644924 IC50 = 15848.93 nM T63414 CX53OM 11652648 IC50 = 15.85 nM T63414 CIQ8C9 11652729 IC50 = 158.49 nM T63414 CJ0X3H 11652890 IC50 = 16.6 nM T63414 CC3ZM8 11653349 IC50 = 19.95 nM T63414 C94XDM 11658739 IC50 = 31622.78 nM T63414 CS3NX6 11681068 IC50 = 3981.07 nM T63414 CJQ19F 11687741 IC50 = 251.19 nM T63414 CXVQ78 11688382 IC50 = 630.96 nM T63414 CA1WS3 11690372 IC50 = 316.23 nM T63414 C7KP6B 11709854 IC50 = 50.12 nM T63414 C90UBJ 11709955 IC50 = 29.51 nM T63414 C45DFS 11744510 IC50 = 19 nM T63414 CC1US4 11749459 IC50 = 110 nM T63414 CN7CG3 11955514 IC50 = 199.53 nM T63414 CKX64A 11955519 IC50 = 190.55 nM T63414 C9YON1 11955520 IC50 = 141.25 nM T63414 CG81BJ 11955559 IC50 = 70.79 nM T63414 C8HW3J 11955560 IC50 = 52.48 nM T63414 C2MTY1 11955601 IC50 = 5.012 nM T63414 CGZ2U6 11955602 IC50 = 51.29 nM T63414 CCXO04 11955641 IC50 = 18.62 nM T63414 C8C1AH 11955642 IC50 = 1380.38 nM T63414 C8O6QT 11955678 IC50 = 57.54 nM T63414 CU5K7B 11955729 IC50 = 147.91 nM T63414 CX1KH4 11955771 IC50 = 407.38 nM T63414 CCPW09 11955827 IC50 = 173.78 nM T63414 CL96MS 11955828 IC50 = 11.75 nM T63414 CZU83X 11955880 IC50 = 131.83 nM T63414 CYC20M 11955881 IC50 = 70.79 nM T63414 C03GKP 11955920 IC50 = 33.88 nM T63414 CYR86X 11955922 IC50 = 34.67 nM T63414 C36WME 11955924 IC50 = 977.24 nM T63414 CPB15O 11955955 IC50 = 39.81 nM T63414 CL04FO 11955956 IC50 = 323.59 nM T63414 CSH71O 11955960 IC50 = 57.54 nM T63414 CXW68G 15486611 IC50 = 31 nM T63414 CX35SR 16678189 IC50 = 15.14 nM T63414 CZB32K 16678190 IC50 = 9.12 nM T63414 CHCM09 16678191 IC50 = 9.12 nM T63414 CVK63O 16678192 IC50 = 11.75 nM T63414 CF2UJ3 16678193 IC50 = 46.77 nM T63414 CE9Q6C 16678194 IC50 = 13.8 nM T63414 CK02CP 16678286 IC50 = 131.83 nM T63414 CD3S5H 16678288 IC50 = 190.55 nM T63414 CD96XF 16678386 IC50 = 190.55 nM T63414 CN14JM 16678387 IC50 = 77.62 nM T63414 COZ8V3 16678388 IC50 = 1047.13 nM T63414 CTF12U 16678389 IC50 = 13182.57 nM T63414 C69EPC 16678391 IC50 = 131.83 nM T63414 C2CNW4 16678483 IC50 = 48.98 nM T63414 CS6M5H 16678489 IC50 = 26.92 nM T63414 CJ2B6L 16678585 IC50 = 1288.25 nM T63414 CE9D7B 16678586 IC50 = 8912.51 nM T63414 CDK64U 16678694 IC50 = 58.88 nM T63414 CJ24DA 16678804 IC50 = 302 nM T63414 CVIU19 16678805 IC50 = 30.9 nM T63414 CUG98F 16678806 IC50 = 48.98 nM T63414 CY3AP8 16678807 IC50 = 19.95 nM T63414 CMKX09 16678903 IC50 = 57.54 nM T63414 C3HF2P 16678904 IC50 = 208.93 nM T63414 CZ39HD 16679400 IC50 = 15.85 nM T63414 CP42YQ 16679489 IC50 = 32.36 nM T63414 C48DST 16679490 IC50 = 67.61 nM T63414 CX20DE 16679491 IC50 = 10.96 nM T63414 C40AYD 16679493 IC50 = 354.81 nM T63414 C7QWN9 16679494 IC50 = 28.84 nM T63414 C09NSJ 16679590 IC50 = 30.9 nM T63414 CQ52JL 16679594 IC50 = 19.05 nM T63414 CIHK17 16679595 IC50 = 50.12 nM T63414 CZ6DV3 16679685 IC50 = 12.59 nM T63414 C9BE2D 16679686 IC50 = 28.18 nM T63414 C3IX1S 16748139 IC50 = 60 nM T63414 CK1C9G 16748140 IC50 > 1000 nM T63414 C9C6DJ 16748141 IC50 > 1000 nM T63414 C52NZH 16748261 IC50 > 1000 nM T63414 CX71LS 16748262 IC50 > 1000 nM T63414 CBAM38 16748263 IC50 > 1000 nM T63414 CHE60A 16748264 IC50 = 12.1 nM T63414 C0FR5J 16748265 IC50 > 1000 nM T63414 CR0E9D 16748266 IC50 > 1000 nM T63414 C1WU4K 16748384 IC50 > 1000 nM T63414 CWJT79 16748385 IC50 > 1000 nM T63414 C9Y7IB 16748386 IC50 > 1000 nM T63414 CTP6G1 16748387 IC50 > 1000 nM T63414 C5I0CX 16748388 IC50 > 1000 nM T63414 C5H8YP 16748389 IC50 > 1000 nM T63414 C10DVY 16748517 IC50 > 1000 nM T63414 CFM3I6 16748518 IC50 > 1000 nM T63414 CEMJ08 16748519 IC50 > 1000 nM T63414 CF3NI1 16748520 IC50 > 1000 nM T63414 CEX26A 16748521 IC50 = 130 nM T63414 CR4K2L 16748522 IC50 > 1000 nM T63414 CU1N4Z 16748628 IC50 > 1000 nM T63414 CID4T1 16748629 IC50 = 40.2 nM T63414 C64BCT 16748630 IC50 > 1000 nM T63414 C25LUG 16748631 IC50 > 1000 nM T63414 CJ9T3Q 16748632 IC50 > 1000 nM T63414 CGPI14 16748633 IC50 = 19.95 nM T63414 C05XNW 16748739 IC50 > 1000 nM T63414 CAKU80 16748740 IC50 = 800 nM T63414 C85QSE 16748741 IC50 > 1000 nM T63414 C4ZAP3 16748742 IC50 > 1000 nM T63414 CWK92R 16748743 IC50 = 35.1 nM T63414 C2Z9YL 16748744 IC50 = 900 nM T63414 CAG01I 16748850 IC50 = 39.81 nM T63414 C9N1AT 16748851 IC50 > 1000 nM T63414 C4Z1DH 16749266 IC50 > 1000 nM T63414 CX1F0R 16749371 IC50 > 1000 nM T63414 C6EM0D 16749372 IC50 = 90.2 nM T63414 CS69QB 16749373 IC50 > 1000 nM T63414 C7XE5Z 16749374 IC50 = 100 nM T63414 CHP82C 16749375 IC50 > 1000 nM T63414 CVH87I 16749376 IC50 > 1000 nM T63414 C0YM8U 18438679 IC50 = 238 nM T63414 C4WP3N 18438683 IC50 = 266 nM T63414 CQG7A5 18438690 IC50 = 95 nM T63414 CG0ZC7 18438692 IC50 = 280 nM T63414 C1Y2TM 18438700 IC50 = 490 nM T63414 C5OPF8 19796304 IC50 = 1 nM T63414 C2KI6R 20173059 IC50 = 2420 nM T63414 C3D9MI 20660005 IC50 = 63.1 nM T63414 C2YI9L 20660020 IC50 = 5.012 nM T63414 C3DT0V 20968164 IC50 = 316.23 nM T63414 CD8CM9 21093784 IC50 = 940 nM T63414 C9BJ7T 21093792 IC50 = 1300 nM T63414 CYA5O7 21093813 IC50 = 1100 nM T63414 C90NZQ 21093814 IC50 = 3600 nM T63414 C0BMP1 21093816 IC50 = 2800 nM T63414 C05FAL 21093905 IC50 = 794.33 nM T63414 COB7R6 22341299 IC50 = 50.12 nM T63414 CVF35Z 22644568 IC50 <= 31622.78 nM T63414 CP6F7H 22644657 IC50 <= 31622.78 nM T63414 CGU0Q2 22644665 IC50 <= 31622.78 nM T63414 C3GVJ2 23649368 IC50 = 132 nM T63414 CK76FP 23649427 Ki = 3.1 nM T63414 C49XAU 23654641 IC50 = 15.85 nM T63414 CC7H0G 23654661 IC50 = 630.96 nM T63414 C47PTE 23654663 IC50 = 251.19 nM T63414 CG39XH 23654666 IC50 = 7.943 nM T63414 C2PV0A 23654747 IC50 = 158.49 nM T63414 CSF46T 23654751 IC50 = 158.49 nM T63414 C1JEP4 23654752 IC50 = 39.81 nM T63414 C73PFO 23654815 IC50 = 2.512 nM T63414 CADC51 23654831 IC50 = 63.1 nM T63414 CKW05E 23654832 IC50 < 3162.28 nM T63414 C5NI0H 23654834 IC50 = 2.512 nM T63414 C5R2VB 24760653 IC50 = 1.995 nM T63414 C2QA6E 24760968 IC50 = 6.31 nM T63414 CMIJ42 24864649 IC50 = 11.48 nM T63414 CZ14WI 24864650 IC50 = 218.78 nM T63414 C6G7YS 24864651 IC50 = 33.88 nM T63414 CET91X 24865007 IC50 = 371.54 nM T63414 CXY74N 24865008 IC50 = 831.76 nM T63414 CRUS91 24865188 IC50 = 38.9 nM T63414 CZF70G 24883277 IC50 > 10000 nM T63414 CEH1K6 24894837 IC50 = 0.1995 nM T63414 C61OTM 24894840 IC50 = 0.05012 nM T63414 CV6B2Z 25011821 IC50 = 3.162 nM T63414 CFB7R4 25014313 IC50 = 0.01 nM T63414 CLA64S 25020193 IC50 = 15.85 nM T63414 C8Y2DG 25022679 IC50 > 10000 nM T63414 CC54IX 25022680 IC50 = 59 nM T63414 C4I6OJ 25032957 IC50 = 34 nM T63414 C68WHE 25061571 IC50 = 10 nM T63414 C39WZD 25061573 IC50 = 10 nM T63414 CZ8S3D 25106221 IC50 = 39.81 nM T63414 C1FER2 25106484 IC50 = 25.12 nM T63414 COEG07 25106658 IC50 = 316.23 nM T63414 C5RC1L 25106660 IC50 = 158.49 nM T63414 CM23AC 25106741 IC50 = 316.23 nM T63414 CPD29L 25106743 IC50 = 63.1 nM T63414 CFN59X 25106744 IC50 = 100 nM T63414 CQC4D9 25107017 IC50 = 50.12 nM T63414 CPJ30M 25107453 IC50 > 630.96 nM T63414 CLIZ02 25159047 IC50 = 28 nM T63414 CT78IL 25210349 IC50 = 31.62 nM T63414 C5F2OH 25809478 IC50 = 3981.07 nM T63414 C3LD7V 40075164 IC50 = 5950 nM T63414 COK46N 44139106 IC50 = 31.62 nM T63414 CJ4QG2 44139223 IC50 = 199.53 nM T63414 C6N8ZH 44139224 IC50 = 251.19 nM T63414 CEGZ59 44139225 IC50 = 251.19 nM T63414 CB0ZD7 44139226 IC50 = 316.23 nM T63414 CD3OL6 44139227 IC50 = 794.33 nM T63414 CZF1I8 44139348 IC50 = 3162.28 nM T63414 CDAY27 44139349 IC50 = 251.19 nM T63414 CA6Q9T 44139350 IC50 = 31622.78 nM T63414 CR19DY 44139351 IC50 = 5011.87 nM T63414 CMYX63 44139352 IC50 = 199.53 nM T63414 CJW89G 44139353 IC50 = 10 nM T63414 CRS4D7 44139469 IC50 = 1995.26 nM T63414 C97IUM 44139470 IC50 = 199.53 nM T63414 C9J4WA 44139598 IC50 = 100 nM T63414 CZ2Q7I 44139724 IC50 = 158.49 nM T63414 C47RUK 44139725 IC50 = 199.53 nM T63414 C9WD4T 44139726 IC50 = 251.19 nM T63414 CHS4Z6 44139727 IC50 = 316.23 nM T63414 C6WFB9 44139728 IC50 = 398.11 nM T63414 CK32IJ 44139877 IC50 = 1000 nM T63414 CJO78K 44139878 IC50 = 1584.89 nM T63414 CRLO92 44139879 IC50 = 794.33 nM T63414 CDM84Y 44139880 IC50 = 2511.89 nM T63414 C87ZUF 44139881 IC50 = 7943.28 nM T63414 C3H6PM 44139882 IC50 = 398.11 nM T63414 C9VJB2 44140001 IC50 = 630.96 nM T63414 CF7RH1 44140002 IC50 = 31.62 nM T63414 CE9WA1 44180167 IC50 = 310 nM T63414 CC14MU 44180168 IC50 = 250 nM T63414 CD51AN 44180169 IC50 = 180 nM T63414 C19ZDA 44241649 IC50 = 4310 nM T63414 CMH56F 44250460 IC50 = 19.95 nM T63414 CB91UW 44352797 IC50 < 10000 nM T63414 CD5MN7 44352798 IC50 = 630.96 nM T63414 C1RV2U 44352806 IC50 = 10000 nM T63414 CVZ85O 44352829 IC50 < 10000 nM T63414 C6FK0N 44352831 IC50 = 630.96 nM T63414 C7S4NI 44352852 IC50 = 6309.57 nM T63414 CW7O4M 44352866 IC50 < 10000 nM T63414 CGI63Q 44352867 IC50 < 10000 nM T63414 CIYE20 44352908 IC50 < 10000 nM T63414 CLR60K 44352910 IC50 < 10000 nM T63414 CNQ8Y9 44352911 IC50 < 10000 nM T63414 CN2RD8 44352912 IC50 < 10000 nM T63414 C3OY6E 44352913 IC50 < 10000 nM T63414 CF24SK 44352947 IC50 = 79.43 nM T63414 CYQ4A7 44352996 IC50 = 125.89 nM T63414 C3CUK0 44353025 IC50 = 158.49 nM T63414 C7D9EM 44353041 IC50 = 158.49 nM T63414 C9HGY8 44353139 IC50 = 199.53 nM T63414 CQ46IG 44353592 EC50 = 52000 nM T63414 CXM4D2 44374511 IC50 = 316 nM T63414 CAN0B9 44388794 IC50 = 63.1 nM T63414 CZ17CH 44388802 IC50 = 125.89 nM T63414 C57VAP 44388827 IC50 > 1000 nM T63414 CXUJ85 44388935 IC50 = 316.23 nM T63414 CH73BF 44388973 IC50 = 79.43 nM T63414 CRKP03 44388975 IC50 = 79.43 nM T63414 CPUT83 44389013 IC50 = 63.1 nM T63414 CMCQ81 44389040 IC50 > 3162.28 nM T63414 C5R3HZ 44391901 IC50 = 79.43 nM T63414 C50EJN 44412196 IC50 > 10000 nM T63414 CO3A0B 44440425 IC50 = 524.81 nM T63414 CT83UQ 44440428 IC50 = 602.56 nM T63414 COEL10 44440430 IC50 = 426.58 nM T63414 CIP1J7 44440432 IC50 = 1819.7 nM T63414 CV6IR5 44440433 IC50 = 6025.6 nM T63414 C1ZO2R 44440436 IC50 = 117.49 nM T63414 CV9W5I 44440439 IC50 = 144.54 nM T63414 C8K9MP 44440442 IC50 = 47.86 nM T63414 C3KF9Q 44440446 IC50 = 48.98 nM T63414 C26ZEO 44440449 IC50 = 912.01 nM T63414 C0YN6I 44440452 IC50 = 213.8 nM T63414 CCL5V1 44440456 IC50 = 331.13 nM T63414 COGQ18 44440459 IC50 = 138.04 nM T63414 CJ0N5Z 44446289 IC50 = 219 nM T63414 CYV62I 44446290 IC50 = 599 nM T63414 C70DYF 44446291 IC50 = 260 nM T63414 CB8SW5 44446292 IC50 = 256 nM T63414 CY5W3J 44446293 IC50 = 504 nM T63414 C9YWH1 44446294 IC50 = 1360 nM T63414 C4I1SC 44446295 IC50 = 539 nM T63414 CJ15XN 44446298 IC50 = 2010 nM T63414 CZXK03 44446299 IC50 = 724 nM T63414 C9Y0VR 44446300 IC50 = 319 nM T63414 CT9R6N 44446317 IC50 = 481 nM T63414 C4LCZ1 44446318 IC50 = 5880 nM T63414 CE0JT5 44446319 IC50 = 517 nM T63414 CDJM56 44446320 IC50 = 3540 nM T63414 C39KPW 44446321 IC50 = 780 nM T63414 C39MDY 44446322 IC50 = 725 nM T63414 CVS3W2 44446323 IC50 = 2460 nM T63414 CZ6J0T 44446324 IC50 = 1540 nM T63414 CP3R2U 44446325 IC50 = 861 nM T63414 C58XIQ 44446327 IC50 = 40 nM T63414 C9JP6I 44453720 IC50 = 67.61 nM T63414 C78FNH 44453771 IC50 = 45.71 nM T63414 CWZ92N 44453795 IC50 = 1621.81 nM T63414 CBA61W 44453817 IC50 = 288.4 nM T63414 CER54H 44453839 IC50 = 20.89 nM T63414 C46EXZ 44453840 IC50 = 154.88 nM T63414 CX5CV8 44453841 IC50 = 478.63 nM T63414 C6PAB1 44453843 IC50 = 47.86 nM T63414 CT3SA5 44453866 IC50 = 616.6 nM T63414 C14RXQ 44453867 IC50 = 3388.44 nM T63414 C7L6BX 44453869 IC50 = 102.33 nM T63414 C7O5BW 44453870 IC50 = 1862.09 nM T63414 CRM84K 44453893 IC50 = 363.08 nM T63414 CP76NZ 44453894 IC50 = 17.78 nM T63414 CSH25Q 44453895 IC50 = 45.71 nM T63414 CZC02W 44454976 IC50 = 140 nM T63414 CTH0Y1 44454978 IC50 = 51 nM T63414 C9DI8L 44454979 IC50 = 88 nM T63414 CZB07S 44455002 IC50 = 58 nM T63414 C4UJE8 44455036 IC50 = 190 nM T63414 C61QTH 44455104 IC50 = 220 nM T63414 CM0Q3T 44455110 IC50 = 430 nM T63414 C4GEW6 44455183 IC50 = 1300 nM T63414 CV9L8T 44455230 IC50 = 460 nM T63414 CG2BU3 44455253 IC50 = 70 nM T63414 CILG68 44455273 IC50 = 57 nM T63414 C2CW5X 44455277 IC50 = 94 nM T63414 CRQ15X 44455311 IC50 = 100 nM T63414 CSV9Z2 44455312 IC50 = 1500 nM T63414 C9BXO1 44455345 IC50 = 1000 nM T63414 CF3MU9 44455378 IC50 = 40 nM T63414 C8S4DG 44455380 IC50 = 60 nM T63414 C3Y2UZ 44455397 IC50 = 110 nM T63414 CXVM85 44455398 IC50 = 71 nM T63414 C7IKG2 44455425 IC50 = 46 nM T63414 CE9VI7 44455448 IC50 = 410 nM T63414 C2B3HJ 44455452 IC50 = 46 nM T63414 CPY02X 44455453 IC50 = 36 nM T63414 COWX27 44455454 IC50 = 40 nM T63414 CEUW63 44455455 IC50 = 310 nM T63414 CJOC69 44567813 IC50 = 25 nM T63414 CE2LB5 44567814 IC50 = 1030 nM T63414 C84VNX 44567815 IC50 = 540 nM T63414 CAH7Z4 44567845 IC50 > 10000 nM T63414 C5OVW0 44567848 IC50 = 780 nM T63414 CYF1R5 44567880 IC50 = 60 nM T63414 CB9SK6 44567881 IC50 = 112 nM T63414 C7FPK6 44567882 IC50 = 40 nM T63414 CQ2CU7 44567883 IC50 = 67 nM T63414 C10QEB 44567914 IC50 = 45 nM T63414 C0MIV1 44567915 IC50 = 130 nM T63414 CWY8Z4 44567916 IC50 = 250 nM T63414 CWP2D0 44567917 IC50 = 24900 nM T63414 CXYI51 44567972 IC50 = 480 nM T63414 C12TOE 44567973 IC50 = 1660 nM T63414 CZ0Q9L 44567974 IC50 = 1330 nM T63414 CJO97Q 44567975 IC50 = 60 nM T63414 CS2YF1 44568011 IC50 = 110 nM T63414 CPG8J6 44568014 IC50 = 93 nM T63414 CX9FB2 44571409 IC50 = 2660 nM T63414 C83OUL 44571411 IC50 = 4410 nM T63414 CR9N4X 44571929 IC50 = 440 nM T63414 C1RF3V 44571930 IC50 = 420 nM T63414 C29IPU 44571977 IC50 = 260 nM T63414 CJX40Z 44571979 IC50 = 400 nM T63414 C1LP0O 44571981 IC50 = 1120 nM T63414 CYX8R0 44572018 IC50 = 5020 nM T63414 C9QAH4 44572020 IC50 = 2560 nM T63414 CNK6G2 44572022 IC50 = 5400 nM T63414 CC5E4B 44572069 IC50 = 820 nM T63414 CZ87DW 44572070 IC50 = 420 nM T63414 C2NW7D 44572072 IC50 = 730 nM T63414 C87PRC 44572124 IC50 = 1530 nM T63414 CJM0C8 44572126 IC50 = 170 nM T63414 C8VO6R 44572127 IC50 = 1260 nM T63414 CGC93W 44572128 IC50 = 2600 nM T63414 CZ3MQ2 44572130 IC50 = 2810 nM T63414 C78EIN 44572132 IC50 = 3220 nM T63414 CAKV23 44576800 IC50 = 27.54 nM T63414 C3TK7V 44576833 IC50 < 1 nM T63414 CE12IZ 44576834 IC50 = 22.91 nM T63414 CRI8B3 44576835 IC50 = 275.42 nM T63414 C4C1FB 44576871 IC50 = 27.54 nM T63414 CX6EC5 45123697 IC50 = 50.12 nM T63414 CQJ49O 45267133 IC50 = 25.12 nM T63414 C9EM1X 45267162 IC50 = 15.85 nM T63414 CFE72S 45267185 IC50 = 501.19 nM T63414 CIF7D9 45267968 IC50 = 10 nM T63414 C48NUE 45269693 IC50 = 7.943 nM T63414 C92BPO 45269772 IC50 > 10000 nM T63414 CRYJ65 45270525 IC50 = 199.53 nM T63414 CG6A1U 45270543 IC50 = 0.3162 nM T63414 CJG3R6 45270588 IC50 = 19.95 nM T63414 C7GD3S 45271344 IC50 <= 10000 nM T63414 CC6UN5 45271415 IC50 > 10000 nM T63414 CA6DH8 45272316 IC50 > 10000 nM T63414 C2NOZ0 45273093 IC50 = 398.11 nM T63414 C8FBV6 45273094 IC50 <= 10000 nM T63414 C7C8SV 45273191 IC50 < 31622.78 nM T63414 C0RVP9 45486014 IC50 = 790 nM T63414 C1T6IN 45486047 IC50 = 13000 nM T63414 CZ0B3A 45486077 IC50 = 1450 nM T63414 CU3H1X 45486078 IC50 = 1280 nM T63414 CJ7R8B 45486080 IC50 = 1180 nM T63414 C3RF4L 45486083 IC50 = 740 nM T63414 CHW0Q6 45486085 IC50 = 850 nM T63414 C2LU4C 45486086 IC50 = 520 nM T63414 CI5G0S 45486088 IC50 = 1420 nM T63414 CG9OH1 45486091 IC50 = 1070 nM T63414 CBPD97 46175179 IC50 > 10000 nM T63414 C80DAS 46231312 IC50 > 10000 nM T63414 C6LJC9 46700791 IC50 = 251.19 nM T63414 C1I6PO 46830282 IC50 = 16 nM T63414 CM6L0H 46830291 IC50 = 27 nM T63414 C01TIE 46831210 IC50 = 33 nM T63414 CYJ24N 46831211 IC50 = 9 nM T63414 CLQ0S5 46831213 IC50 = 39 nM T63414 C2W8ID 46832336 IC50 = 23 nM T63414 CPE2Z1 46834939 IC50 = 104 nM T63414 CT2AE5 46834941 IC50 = 92 nM T63414 CHP14S 46834942 IC50 = 38 nM T63414 CA06XH 46886951 IC50 = 32 nM T63414 C7QL1Y 46886952 IC50 = 449 nM T63414 C5L3VP 46886953 IC50 = 17 nM T63414 CR2P7T 46886954 IC50 = 46 nM T63414 CU16JH 46886955 IC50 = 51 nM T63414 C46RHT 46887106 IC50 = 125.89 nM T63414 CTIN74 46887107 IC50 > 1000 nM T63414 C0UK6V 46887108 IC50 > 1000 nM T63414 CE13QO 46887141 IC50 > 1000 nM T63414 C7AID1 46887142 IC50 > 1000 nM T63414 CV1XW4 46887143 IC50 = 251.19 nM T63414 CDUO76 46887144 IC50 > 1000 nM T63414 CT6LC8 46887145 IC50 = 158.49 nM T63414 C0IZ2X 46887191 IC50 = 158.49 nM T63414 CFKC73 46887193 IC50 > 1000 nM T63414 CJB92T 46887194 IC50 > 1000 nM T63414 CLW5I3 46887195 IC50 > 1000 nM T63414 C3E4LZ 46887223 IC50 = 39.81 nM T63414 C9MO4K 46887224 IC50 = 10 nM T63414 CWC97Y 46887252 IC50 = 125.89 nM T63414 C9NFM0 46887253 IC50 = 199.53 nM T63414 CCZ9I6 46887477 IC50 = 40 nM T63414 CS0K7X 46887514 IC50 = 213 nM T63414 CLF08T 46887515 IC50 = 134 nM T63414 CCU0J8 46887516 IC50 = 232 nM T63414 C4LN5B 46887517 IC50 = 17 nM T63414 CD5F4G 46887518 IC50 = 32 nM T63414 C6TPL2 46887560 IC50 = 56 nM T63414 CM58OE 46887561 IC50 = 18 nM T63414 CBPU74 46887562 IC50 = 22 nM T63414 C1WBI0 46887563 IC50 = 8 nM T63414 CLV1W2 46918487 IC50 = 39.81 nM T63414 CY1OI8 49803437 IC50 = 932 nM T63414 CR1W5M 49863038 IC50 = 10 nM T63414 CLDK29 49863078 IC50 = 125.89 nM T63414 CH18IF 49863079 IC50 = 100 nM T63414 CGXC76 49863080 IC50 = 158.49 nM T63414 C5XZN3 49863081 IC50 > 1000 nM T63414 CW7Z8Q 49863082 IC50 = 12.59 nM T63414 C02NHY 49863083 IC50 = 398.11 nM T63414 CL45EU 49863107 IC50 = 158.49 nM T63414 CQN7K5 49863108 IC50 = 316.23 nM T63414 CE8FN5 49863109 IC50 = 63.1 nM T63414 CEB9H4 49864819 IC50 = 501.19 nM T63414 CPQ0C5 49864874 IC50 = 794.33 nM T63414 CY1NP4 49864875 IC50 = 100 nM T63414 CFWJ63 49864876 IC50 < 1000 nM T63414 CQ7K6V 49864877 IC50 = 100 nM T63414 C1VJ3X 49864911 IC50 = 31.62 nM T63414 CCN40K 49864912 IC50 = 158.49 nM T63414 CKBY67 49864913 IC50 = 398.11 nM T63414 CKTJ85 49864914 IC50 < 1000 nM T63414 CR0M7Y 49864915 IC50 = 25.12 nM T63414 CTV2R6 49864916 IC50 < 1000 nM T63414 C8Q0IP 49864946 IC50 < 1000 nM T63414 CNA3I9 49864947 IC50 = 79.43 nM T63414 C3VU2Y 49864948 IC50 = 630.96 nM T63414 CFT3V8 49864949 IC50 < 1000 nM T63414 CO1Y8A 49864950 IC50 = 630.96 nM T63414 C6Q5PX 49864951 IC50 = 100 nM T63414 C8Y0QK 49864952 IC50 = 630.96 nM T63414 CA1ZP4 49865005 IC50 < 1000 nM T63414 C9VB5R 49865006 IC50 = 12.59 nM T63414 CEQ42N 49865007 IC50 = 6.31 nM T63414 C9TX8W 49865008 IC50 = 1.585 nM T63414 CPO7N8 49865009 IC50 < 1000 nM T63414 CVLW35 49865010 IC50 = 100 nM T63414 CM3R5F 49865011 IC50 < 1000 nM T63414 CE93YS 49865054 IC50 = 158.49 nM T63414 C5UJL2 49865055 IC50 = 31.62 nM T63414 C0S2UE 50898450 IC50 = 10 nM T63414 C8P3FI 52543399 IC50 = 6410 nM T63414 CD52NL 52940698 IC50 = 3.981 nM T63414 CD4YE2 52941885 IC50 = 3.981 nM T63414 C7NV6R 52942125 IC50 = 31.62 nM T63414 C60DON 52943044 IC50 = 1.995 nM T63414 C3YWI6 52943045 IC50 = 10 nM T63414 CS46RU 52943071 IC50 = 5.012 nM T63414 CBRT15 52943107 IC50 = 79.43 nM T63414 CQ0B4W 52943108 IC50 = 25.12 nM T63414 CO9X7I 52943116 IC50 = 2.512 nM T63414 CYJ72M 52944502 IC50 = 0.631 nM T63414 CPG4J9 52944504 IC50 = 3.981 nM T63414 CM72WO 52946486 IC50 = 10 nM T63414 CC29MO 52946708 IC50 = 25.12 nM T63414 CWV76B 52947925 IC50 = 25.12 nM T63414 C78WQD 52947971 IC50 = 3.981 nM T63414 CDVR73 52949177 IC50 = 10 nM T63414 CM7B8F 53248666 IC50 = 14.79 nM T63414 C87LRM 53249126 IC50 = 11.48 nM T63414 C4KJN3 53357190 IC50 = 50 nM T63414 CFNV60 53357191 IC50 = 29 nM T63414 CV4NJ5 53357192 IC50 = 24 nM T63414 C3HO2R 53388310 IC50 = 3 nM T63414 C5BQU3 53388312 IC50 = 0.5 nM T63414 CG1L4T 54580621 IC50 = 64 nM T63414 CNI84W 54580632 IC50 = 41 nM T63414 C2OP1Q 54580633 IC50 = 132 nM T63414 CZJ87H 54580659 IC50 = 13.8 nM T63414 C3OZE5 54580660 IC50 = 21.88 nM T63414 C3RAB9 54580661 IC50 = 120.23 nM T63414 CE68YQ 54580681 IC50 = 74.13 nM T63414 CB7S6Y 54580682 IC50 = 54.95 nM T63414 CD9R1X 54580683 IC50 = 26.92 nM T63414 CWH45G 54581536 IC50 > 5000 nM T63414 CQW6Y4 54581643 IC50 = 25 nM T63414 CAF1W3 54581644 IC50 = 41 nM T63414 C9NYE7 54581645 IC50 = 64 nM T63414 CZB03V 54581673 IC50 = 16.6 nM T63414 C72LDF 54581674 IC50 = 27.54 nM T63414 CKVL16 54581675 IC50 = 82 nM T63414 CBT56Y 54581676 IC50 = 248 nM T63414 CJ82ZY 54581694 IC50 = 562.34 nM T63414 C90TNZ 54581695 IC50 = 1905.46 nM T63414 CUSK31 54581696 IC50 = 14.79 nM T63414 C4WJP0 54582634 IC50 = 141 nM T63414 C4OQ0E 54582635 IC50 = 470 nM T63414 C3M7BF 54582636 IC50 = 3207 nM T63414 C0MV6O 54582637 IC50 = 1236 nM T63414 CO6T7E 54582658 IC50 = 23.99 nM T63414 C5YMS4 54582659 IC50 = 43 nM T63414 C31HVQ 54582660 IC50 = 51 nM T63414 CEQK29 54582681 IC50 = 436.52 nM T63414 CO78WU 54582682 IC50 = 5623.41 nM T63414 CA35XM 54583586 IC50 = 121 nM T63414 C9E2DV 54583587 IC50 = 36 nM T63414 CL9HZ2 54583588 IC50 = 52 nM T63414 CZ36RH 54583589 IC50 = 439 nM T63414 CUIL26 54583619 IC50 = 40.74 nM T63414 CW6M0F 54583620 IC50 = 31.62 nM T63414 CC4ZP6 54583646 IC50 = 28.18 nM T63414 CB3N6C 54583647 IC50 = 38.9 nM T63414 C34SBA 54584488 IC50 = 185 nM T63414 CWV3S2 54584577 IC50 = 4065 nM T63414 C79HIA 54584578 IC50 = 117 nM T63414 CXC2J1 54584579 IC50 = 1471 nM T63414 CU19XD 54584620 IC50 = 74.13 nM T63414 CO5A6J 54584621 IC50 = 19.95 nM T63414 C2J6ED 54584622 IC50 = 70.79 nM T63414 CG7C0N 54584623 IC50 = 87.1 nM T63414 CC8JA2 54585434 IC50 = 42 nM T63414 CC5EH6 54585435 IC50 = 700 nM T63414 CW9AR7 54585517 IC50 = 158 nM T63414 CJ9R3L 54585518 IC50 = 114 nM T63414 C41NMK 54585519 IC50 = 143 nM T63414 CHA0L2 54585520 IC50 = 207 nM T63414 C5MCX8 54585545 IC50 = 39.81 nM T63414 CY3NR0 54585546 IC50 = 31.62 nM T63414 CAJ7W9 54585547 IC50 = 257.04 nM T63414 C7C4OB 54585548 IC50 = 42 nM T63414 CWO7F1 54585568 IC50 = 234.42 nM T63414 CB40QJ 54585569 IC50 = 15.85 nM T63414 CNRW68 54586397 IC50 = 200 nM T63414 C9MJH2 54586491 IC50 = 52 nM T63414 CS79DZ 54586492 IC50 = 111 nM T63414 C01NPQ 54586493 IC50 = 40 nM T63414 C85ZRN 54586494 IC50 = 114 nM T63414 C0E7LC 54586495 IC50 = 73 nM T63414 CXYL81 54586524 IC50 = 18.2 nM T63414 C1FYE9 54587413 IC50 > 5000 nM T63414 C0B5GH 54587523 IC50 = 35 nM T63414 CIL8Y6 54587524 IC50 = 43 nM T63414 C3VWR8 54587525 IC50 = 252 nM T63414 CNBI30 54587526 IC50 = 35 nM T63414 CSU91D 54587578 IC50 = 30.2 nM T63414 C7Y9QF 56589589 IC50 = 24 nM T63414 CW20CN 56658584 IC50 = 250 nM T63414 CA8W3B 56658585 IC50 = 1050 nM T63414 CXW93P 56658695 IC50 = 4800 nM T63414 CN2Y8B 56662034 IC50 = 6 nM T63414 C3X6SW 56662173 IC50 = 1600 nM T63414 CPO39Q 56662911 IC50 = 50.12 nM T63414 CV2IO3 56662912 IC50 = 158.49 nM T63414 CXF5Q2 56662950 IC50 = 199.53 nM T63414 C1HT4M 56665515 IC50 = 720 nM T63414 C0SN9Z 56665516 IC50 = 510 nM T63414 C3ZR5Q 56666388 IC50 = 50.12 nM T63414 CQE0H2 56666425 IC50 = 100 nM T63414 CNI50D 56666426 IC50 = 31.62 nM T63414 CJ6SG0 56666427 IC50 = 39.81 nM T63414 CS49UN 56668947 IC50 = 460 nM T63414 CT7SK3 56668948 IC50 = 240 nM T63414 C8JF5B 56669848 IC50 = 50.12 nM T63414 CZ0JP1 56672431 IC50 = 4600 nM T63414 C8WEG7 56675816 IC50 = 5200 nM T63414 CXW23S 56676617 IC50 = 100 nM T63414 C87VZL 56676618 IC50 = 50.12 nM T63414 CQV48D 56676619 IC50 = 50.12 nM T63414 C2SW4X 56679127 IC50 = 668 nM T63414 CJMO40 56679990 IC50 = 125.89 nM T63414 CQYN10 56679991 IC50 = 63.1 nM T63414 C2BQ9G 56683282 IC50 = 100 nM T63414 CEP6F0 56683327 IC50 = 63.1 nM T63414 C4LQK6 56683328 IC50 = 501.19 nM T63414 C9KI8H 57390667 IC50 = 50 nM T63414 CH6J9B 57392463 IC50 = 101 nM T63414 C5ZCB2 57392464 IC50 = 28 nM T63414 CQ5HO4 57392465 IC50 = 45 nM T63414 C9TLV4 57392466 IC50 = 1944 nM T63414 C8DE7B 57394171 IC50 = 388 nM T63414 CBAH26 57394172 IC50 = 276 nM T63414 CBMW74 57394173 IC50 = 700 nM T63414 C6WP2N 57394174 IC50 = 91 nM T63414 CF9NK7 57394175 IC50 = 52 nM T63414 CAJE41 57394176 IC50 = 39 nM T63414 CC4D5S 57394312 IC50 = 178 nM T63414 C0LX4E 57394313 IC50 = 85 nM T63414 C0NS6G 57395953 IC50 = 25 nM T63414 CT4X5P 57397748 IC50 = 110 nM T63414 C39CQX 57399409 IC50 = 108 nM T63414 CA57EW 57399410 IC50 = 104 nM T63414 C0WF7P 57399411 IC50 = 95 nM T63414 CE98JC 57399524 IC50 = 937 nM T63414 CD65TQ 57399525 IC50 = 870 nM T63414 C7S2RH 57399526 IC50 = 107 nM T63414 C4A9HB 57401171 IC50 = 55 nM T63414 CTN6K9 57401282 IC50 = 237 nM T63414 C4DUJ3 57401283 IC50 = 845 nM T63414 C0H2XN 57402932 IC50 = 137 nM T63414 CGH68E 57403034 IC50 = 269 nM T63414 CG1BC2 57403035 IC50 = 1036 nM T63414 C3POX4 57412481 IC50 = 900 nM T63414 CX50UV 57412482 IC50 = 1100 nM T63414 CT6Q4M 57412483 IC50 = 1400 nM T63414 CD6IN7 57412484 IC50 = 1500 nM T63414 CIXG79 57412485 IC50 = 620 nM T63414 C3F0YK 57412486 IC50 = 2500 nM T63414 CQF81U 57412565 IC50 = 1100 nM T63414 CNV98G 57412566 IC50 = 770 nM T63414 CC6BO8 57412567 IC50 = 1200 nM T63414 C84XCU 57412568 IC50 = 1900 nM T63414 C2WI7A 57412569 IC50 = 950 nM T63414 C56ICN 57412570 IC50 = 370 nM T63414 CL2ZY8 57412662 IC50 = 1100 nM T63414 C7ESN1 57412663 IC50 = 4200 nM T63414 CDQL71 57412664 IC50 = 320 nM T63414 CW1V0E 57412668 IC50 = 1200 nM T63414 CFS42I 57412745 IC50 = 380 nM T63414 C26MYQ 57412746 IC50 = 56 nM T63414 C81YML 57412747 IC50 = 42 nM T63414 CA1FY2 57412748 IC50 = 730 nM T63414 CJ7P2M 57412749 IC50 = 360 nM T63414 CV3H5P 57412750 IC50 = 340 nM T63414 CF1RD7 57412751 IC50 = 77 nM T63414 CY0CZ1 57412921 IC50 = 900 nM T63414 C67YRL 58227894 IC50 = 64 nM T63414 C0T1SR 58227950 IC50 = 82 nM T63414 CZEJ87 58228090 IC50 = 85 nM T63414 CT1EL4 58228091 IC50 = 151 nM T63414 CJ9EB3 58228418 IC50 = 78 nM T63414 CRSI26 58228496 IC50 = 120 nM T63414 CJ5Y4X 58228512 IC50 = 35 nM T63414 CS9LM2 59377426 IC50 = 23 nM T63414 CLPY52 59377517 IC50 = 20 nM T63414 C19YVT 59377518 IC50 = 8 nM T63414 C1JK7V 59377559 IC50 = 30 nM T63414 C4CD3N 59377565 IC50 = 27 nM T63414 CK23UQ 59377575 IC50 = 6 nM T63414 CQZ4H9 59377579 IC50 = 17 nM T63414 C24VHF 59377604 IC50 = 33 nM T63414 C0Z9CB 59377671 IC50 = 3800 nM T63414 C5T4CV 59377728 IC50 = 37 nM T63414 C3OY9U 59377733 IC50 = 40 nM T63414 C6GE1D 59377797 IC50 = 32 nM T63414 CHYU80 59377854 IC50 = 9 nM T63414 CDN3P6 59377867 IC50 = 12 nM T63414 CO4N7S 59377977 IC50 = 9 nM T63414 CM4EF3 59378034 IC50 = 9 nM T63414 C49IHZ 59760814 IC50 = 51 nM T63414 CO7PZ5 60168729 IC50 > 10000 nM T63414 C1IW8C 66598994 IC50 = 2.1 nM T63414 CTY7A5 66599177 IC50 = 7.9 nM T63414 C7W6RA 66599198 IC50 = 1.9 nM T63414 CFH6T5 66599261 IC50 < 10 nM T63414 CV6YT7 66599277 IC50 = 9.7 nM T63414 CB2U9J 67460623 Ki = 54.2 nM T63414 C0PK9J 70684134 IC50 = 13 nM T63414 C1XWD2 70690419 IC50 = 1400 nM T63414 CNW4E7 70690420 IC50 = 2800 nM T63414 CZ60JU 70692584 IC50 = 4.9 nM T63414 CL0JG7 70692585 IC50 = 210 nM T63414 C6IE1L 70794829 IC50 = 21 nM T63414 CH9Q0R 71450180 IC50 > 10000 nM T63414 CR64QG 71457337 IC50 > 10000 nM T63414 CR1L5W 71459185 IC50 = 1270 nM T63414 CSV43Z 71459189 IC50 > 10000 nM T63414 C0Y1JN 71462707 IC50 > 10000 nM T63414 CY9HC1 71464744 IC50 = 217 nM T63414 CIV3A7 71464745 IC50 = 666 nM T63414 CXH37V 71464746 IC50 = 220 nM T63414 CA1YJ5 71464747 IC50 = 133 nM T63414 CIU6C4 71464792 IC50 = 913 nM T63414 C31QEJ 71464793 IC50 = 72 nM T63414 CK5X2U 71464795 IC50 = 423 nM T63414 CJD57F 71464849 IC50 = 4880 nM T63414 CEO40G 71465164 IC50 = 3820 nM T63414 CU59BL 71465203 IC50 = 885 nM T63414 CP5CQ4 71465253 IC50 = 1820 nM T63414 CBI48D 71465254 IC50 = 1620 nM T63414 CIJ98Q 71465297 IC50 = 574 nM T63414 CATI79 71465298 IC50 = 789 nM T63414 CQV0T9 71465299 IC50 = 1010 nM T63414 CNUP45 71465300 IC50 = 5730 nM T63414 CH0FQ9 71465345 IC50 = 4990 nM T63414 CL03EH 71465347 IC50 = 11700 nM T63414 CAG4Z9 71465348 IC50 = 5650 nM T63414 C0AMR2 71465349 IC50 = 8770 nM T63414 CP5SD6 71465398 IC50 = 133 nM T63414 C3SWP9 71465399 IC50 = 7220 nM T63414 C6X3UJ 71465489 IC50 = 3760 nM T63414 CF2EL6 71466065 IC50 = 2140 nM T63414 CA65EM 71466067 IC50 = 1200 nM T63414 C4JH5Q 71466147 IC50 = 3430 nM T63414 CTZ90M 71466149 IC50 = 66 nM T63414 C6I0RB 71466213 IC50 = 107 nM T63414 CY5RP0 71466214 IC50 = 12 nM T63414 CQ5M0F 71466215 IC50 = 23 nM T63414 CNKP68 71466216 IC50 = 21 nM T63414 CLV2M3 71466284 IC50 = 131 nM T63414 C0VWJ2 71466285 IC50 = 25 nM T63414 C8C0KV 71466286 IC50 = 17 nM T63414 C60JFN 71466340 IC50 = 664 nM T63414 CUDK53 71466341 IC50 = 583 nM T63414 C4BOQ5 71466342 IC50 = 215 nM T63414 CBOT16 71466343 IC50 = 710 nM T63414 C5SAP9 71466396 IC50 = 30 nM T63414 C9YK3U 71466397 IC50 = 60 nM T63414 CIY5D8 71466398 IC50 = 169 nM T63414 CPV4S3 71466399 IC50 = 99 nM T63414 CNI81D 71466472 IC50 = 32 nM T63414 C5ELV2 71466473 IC50 = 166 nM T63414 C3YA7I 71466474 IC50 = 14 nM T63414 C80BPO 71466475 IC50 = 361 nM T63414 CJPR13 71625847 Ki = 12.59 nM T63414 C3U1YM 73669299 IC50 = 95200 nM T63414 C59FZS 76310220 IC50 = 3981.07 nM T63414 C4VIN2 76313910 IC50 = 3981.07 nM T63414 CB69EX 76324694 IC50 > 100000 nM T63414 C2BE9J 76853227 IC50 = 1.5 nM T63414 CS2N0Z 78153059 IC50 = 1.3 nM T63414 CQMB31 85470872 IC50 = 3.467 nM T63414 CA1CE3 86270720 IC50 = 4 nM T63414 C9TE7X 86271008 IC50 = 15 nM T63414 CMZV56 86271009 Ki = 40 nM T63414 CXN93A 86271108 IC50 = 2.188 nM T63414 C2KHM0 86271111 IC50 = 26 nM T63414 CN9MO7 86271494 IC50 = 4.8 nM T63414 CD6IJ1 86271658 IC50 = 4 nM T63414 CU4H0C 86271659 IC50 = 12 nM T63414 C5LD6M 86271660 IC50 = 89 nM T63414 C6ND4T 86271664 IC50 = 9 nM T63414 CWZ13M 86271758 IC50 = 14 nM T63414 C0D6MG 86271759 IC50 = 5 nM T63414 C3QR6J 86271850 IC50 = 10 nM T63414 CH3I6S 86271851 IC50 = 34 nM T63414 C2PE9L 86271853 IC50 = 78 nM T63414 C87QHD 86271941 IC50 = 9 nM T63414 CY01FH 86271942 IC50 = 30 nM T63414 CS74NP 86279014 IC50 = 6960 nM T63414 CQVL07 86279015 IC50 = 216 nM T63414 C6DX8V 86279088 IC50 = 3.4 nM T63414 C53GEN 86279089 IC50 = 72 nM T63414 C0ST4V 86279091 IC50 = 3.6 nM T63414 C58YOW 86279280 IC50 = 440 nM T63414 CW9KT6 86279350 IC50 = 1 nM T63414 C2NZE7 86279351 IC50 = 3.4 nM T63414 C4HLA3 86279411 IC50 = 4710 nM T63414 C38CMG 86279412 IC50 = 0.7 nM T63414 C5PLE7 86279413 IC50 = 0.2 nM T63414 C1EJ2H 86279414 IC50 = 0.5 nM T63414 CW7VE6 86279479 IC50 = 4.2 nM T63414 C7ETD9 86279481 IC50 = 0.5 nM T63414 C80FHL 86279482 IC50 = 0.6 nM T63414 CA35JQ 86279547 IC50 = 1.9 nM T63414 CR15JV 86279548 IC50 = 0.7 nM T63414 C5OM4Q 86279551 IC50 = 3.8 nM T63414 C8HK2T 86279746 IC50 = 4.3 nM T63414 CPJV10 86280878 IC50 = 19 nM T63414 C9ZS2N 86281547 IC50 = 28.1 nM T63414 C86FUO 86281680 IC50 = 4.5 nM T63414 CE68GI 86281948 IC50 = 240 nM T63414 CC3Z1H 86281949 IC50 = 8.5 nM T63414 CYK2T9 86282366 EC50 = 158 nM T63414 CA74MT 86282635 IC50 = 10 nM T63414 C3AS7V 86716303 IC50 = 0.79 nM T63414 CJ2NE0 88884677 IC50 = 9 nM T63414 CH8JM7 88954244 IC50 = 25 nM T63414 CO8M2K 90407576 Ki = 15.4 nM T63414 CA47VK 90408538 Ki = 22 nM T63414 CTC8B5 90408742 IC50 = 3538 nM T63414 CFG74P 90408756 IC50 = 7.3 nM T63414 CE4IT5 90408860 IC50 = 10 nM T63414 CZB5W4 90408922 IC50 = 880 nM T63414 C3E1CS 90409007 IC50 = 14 nM T63414 C1VA4O 90409557 IC50 = 1.9 nM T63414 C67XEH 90409637 IC50 = 114 nM T63414 CJ6E1S 90409668 IC50 = 28 nM T63414 CJPC93 90410264 IC50 = 1.7 nM T63414 C2FKB3 90410598 IC50 = 8 nM T63414 CB0RP3 90410604 IC50 = 8.318 nM T63414 CQ8ZW3 90410911 IC50 = 5.37 nM T63414 C2ZSD8 90444843 IC50 = 65 nM T63414 CR8KM2 90452359 IC50 = 77 nM T63414 CN9Y7U 90452374 IC50 = 12 nM T63414 C1EVN3 90455889 IC50 = 1.8 nM T63414 CAGK52 90456097 IC50 = 2 nM T63414 C5EC1H 90456171 IC50 = 19 nM T63414 C2JP5R 102004341 IC50 = 4.9 nM T63414 C4YI1F 108870288 IC50 = 3380 nM T63414 C1VF4Q 108870345 IC50 = 6750 nM T63414 CEFX57 117614925 IC50 = 14 nM T63414 CC5H9Y 117614990 IC50 = 11 nM T63414 C73LFS 118001660 IC50 = 809 nM T63414 CC37SU 118001939 IC50 = 810 nM T63414 CF57IP 118289475 IC50 = 18 nM T63414 C1YHC2 118566570 IC50 = 8.2 nM T63414 C9XV8C 118566572 IC50 = 36 nM T63414 C81DBJ 118566586 IC50 = 94 nM T63414 C0Z8PK 118566589 IC50 = 47 nM T63414 C16QEP 118566591 IC50 = 19 nM T63414 CGLB17 118566597 IC50 = 18 nM T63414 CWT5D6 118566606 IC50 = 140 nM T63414 C6VOL1 118566607 IC50 = 37 nM T63414 CCT20R 118566608 IC50 = 72 nM T63414 CSZ90X 118566610 IC50 = 89 nM T63414 C3H4AL 118566616 IC50 < 10 nM T63414 CY8P1K 118566647 IC50 = 27 nM T63414 C8XAS5 118566649 IC50 = 50 nM T63414 COZ29M 118566667 IC50 = 4.5 nM T63414 CM2YC8 118569729 IC50 = 230 nM T63414 CUI9F8 118569766 IC50 = 10 nM T63414 C2YU9O 118733180 IC50 = 14 nM T63414 CC74NF 118733181 IC50 = 12000 nM T63414 CQ5B1O 118733182 IC50 = 8960 nM T63414 C4T6YE 118733183 IC50 = 1970 nM T63414 CD26ZV 118733184 IC50 = 12200 nM T63414 CBI29Y 118733185 IC50 = 7720 nM T63414 CFCN02 118733187 IC50 = 355 nM T63414 CHWJ79 118733188 IC50 = 2290 nM T63414 C8F5WU 118733189 IC50 = 15 nM T63414 C9W3EM 118733190 IC50 = 27 nM T63414 CU5LV0 118733191 IC50 = 81 nM T63414 CPI50J 118733192 IC50 = 49 nM T63414 C03PZR 118733193 IC50 = 29 nM T63414 CVQU96 118733194 IC50 = 50 nM T63414 C69ZDL 118733195 IC50 = 542 nM T63414 CSQ21V 118733196 IC50 = 847 nM T63414 CXN07V 118733197 IC50 = 1670 nM T63414 C19UPL 118733198 IC50 = 3240 nM T63414 CAO73D 118949526 IC50 = 6.9 nM T63414 C79OSH 118949550 IC50 = 14 nM T63414 C7VL6I 118949555 IC50 = 1.4 nM T63414 C2KE6S 118949557 IC50 = 3.9 nM T63414 CN56FH 118949563 IC50 = 7.7 nM T63414 C8XWC1 118949568 IC50 = 15 nM T63414 CKL65X 118949576 IC50 = 23 nM T63414 CZQJ64 118949580 IC50 = 1670 nM T63414 CC3ZQ6 118949582 IC50 = 1560 nM T63414 CC03VS 118949592 IC50 = 12 nM T63414 C9LH2E 118950072 IC50 = 8.2 nM T63414 C7CPN2 118950092 IC50 = 8.7 nM T63414 C2BM9A 118950093 IC50 = 29 nM T63414 C4I2CJ 118950115 IC50 = 2.4 nM T63414 CWR8M4 118950147 IC50 = 7.7 nM T63414 CK74CV 118950157 IC50 = 8 nM T63414 CET0J1 118950171 IC50 = 8.5 nM T63414 CN71LF 118950176 IC50 = 3.2 nM T63414 CR3A8E 118950327 IC50 = 10 nM T63414 CE8G3M 118950384 IC50 = 55 nM T63414 C9UHO7 118950386 IC50 = 6.3 nM T63414 C6GJ2X 118950391 IC50 = 11 nM T63414 C1HJD2 118950410 IC50 = 10 nM T63414 C3GA0C 118950451 IC50 = 8.7 nM T63414 CI9MA2 118950452 IC50 = 12 nM T63414 CP0ZM7 118950460 IC50 = 7 nM T63414 CH5CU4 118950468 IC50 = 2.7 nM T63414 CD13JM 118950470 IC50 = 1370 nM T63414 CCX9B0 118950531 IC50 > 10000 nM T63414 CKG4N5 123779233 IC50 = 875 nM T63414 CPO7N5 124125214 IC50 = 10600 nM T63414 CJ5I8K 125478479 IC50 = 5.3 nM T63414 C68WFZ 127038803 IC50 = 252 nM T63414 CL0Y3F 127040183 IC50 > 10000 nM T63414 CM6QR9 127041723 IC50 = 1000 nM T63414 CD1N6H 127041895 IC50 > 10000 nM T63414 C1Z7PJ 127045201 IC50 = 1156.1 nM T63414 C34KHO 135603818 IC50 = 897 nM T63414 C3K1CM 135960707 IC50 = 6400 nM T63414 C3MR6C 136000710 IC50 = 1253.6 nM T63414 CN1VW6 137632041 IC50 = 18000 nM T63414 C5Q2HE 137632064 IC50 = 1557000 nM T63414 C6KC4F 137632084 IC50 = 389 nM T63414 CZ81QC 137633557 IC50 = 851 nM T63414 CC93IR 137635457 IC50 = 3020 nM T63414 CM6T5X 137635730 IC50 = 138 nM T63414 C0VRU5 137637027 IC50 = 100 nM T63414 CZH73L 137638115 IC50 = 132 nM T63414 CS2X8I 137638643 IC50 = 79 nM T63414 C5AIM2 137638655 IC50 = 186 nM T63414 CV5BE6 137640398 IC50 = 58 nM T63414 CPIG47 137640412 IC50 = 2 nM T63414 C9R8EP 137640871 IC50 = 214 nM T63414 CZ3VP0 137641909 IC50 = 51 nM T63414 CG3ZK6 137644370 IC50 = 933000 nM T63414 C6YO0L 137644636 IC50 = 40 nM T63414 CC3BS8 137646461 IC50 > 10000 nM T63414 CTKZ94 137646544 IC50 = 4034 nM T63414 C7BXL2 137646572 IC50 = 2399 nM T63414 C5GS2K 137646668 IC50 > 10000 nM T63414 CH3T7M 137649164 IC50 > 10000 nM T63414 C3PI9R 137650645 IC50 = 132000 nM T63414 CEJ6I1 137651790 IC50 > 10000 nM T63414 C4X0OY 137652052 IC50 = 366000 nM T63414 CJ2NS6 137652085 IC50 = 96000 nM T63414 C86LNH 137652744 IC50 = 58 nM T63414 CRB7N0 137652989 IC50 = 501 nM T63414 CM34CG 137655633 IC50 > 10000 nM T63414 CI0Q4V 137657140 IC50 > 10000 nM T63414 CKX62S 137658719 IC50 = 562 nM T63414 CNG5A9 137659120 IC50 = 417 nM T63414 CN6C9F 137660086 IC50 = 562 nM T63414 C8IEL0 137660769 IC50 = 4070 nM T63414 CVY90C 137661206 IC50 = 2455 nM T63414 C3JKD5 137661884 IC50 = 174 nM T63414 CRX48H 142737903 IC50 = 27 nM T63414 CGYE15 142737904 IC50 > 10000 nM T63414 CH9TP6 142737905 IC50 = 244 nM T63414 C6J8QD 142737906 IC50 = 702 nM T63414 C2K3ZM 142737910 IC50 = 32 nM T63414 C7PD9T 142737911 IC50 = 249 nM T63414 CW48KL 142737912 IC50 = 3520 nM T63414 C92ATU 142737914 IC50 = 202 nM T63414 CD8ZI3 142737915 IC50 = 312 nM T63414 CZD8J6 142737916 IC50 = 7 nM T63414 CEZ87J 142737917 IC50 = 210 nM T63414 C4TR6I 142737918 IC50 = 565 nM T63414 C5PS0V 142737919 IC50 = 1440 nM T63414 C3PT7Y 142737920 IC50 = 1.49 nM T63414 C43ZJQ 142737921 IC50 > 10000 nM T63414 CUC6I0 142737923 IC50 = 26 nM T63414 CU80EL 142737924 IC50 = 22 nM T63414 CH3X6D 142737925 IC50 > 10000 nM T63414 CPN42E 142737926 IC50 = 259 nM T63414 CST93I 142737929 IC50 = 269 nM T63414 C9SPQ7 142737930 IC50 = 37 nM T63414 CJG4Q0 142737931 IC50 = 400 nM T63414 CO23GR 142737932 IC50 = 0.49 nM T63414 CU78YD 142737933 IC50 = 430 nM T63414 CIC78M 142737934 IC50 = 155 nM T63414 CB42JQ 142737935 IC50 = 896 nM T63414 CGOA34 142737938 IC50 = 64 nM T63414 C35IFV 142737939 IC50 = 13 nM T63414 CY75NU 142737940 IC50 = 0.32 nM T63414 CEOY83 142737941 IC50 > 10000 nM T63414 C0I4TF 142737942 IC50 = 202 nM T63414 C0O4LP 142737943 IC50 = 143 nM T63414 C28KQI 142737944 IC50 = 58 nM T63414 C7B2HO 142737945 IC50 = 13 nM T63414 C3ZOV5 142737950 IC50 = 1.33 nM T63414 C37UNR 142737951 IC50 = 238 nM T63414 C9CLA6 142737953 IC50 = 4.28 nM T63414 C7ZQ4N 142737954 IC50 = 41 nM T63414 CI7P6A 142737955 IC50 = 0.11 nM T63414 CH52OW 142737956 IC50 = 1.76 nM T63414 CG23WO 142737957 IC50 = 152 nM T63414 CB52JH 142737959 IC50 = 187 nM T63414 C8R5LV 142737960 IC50 = 1570 nM T63414 CTK68D 142737961 IC50 = 22 nM T63414 C6WY0F 142737963 IC50 = 4.7 nM T63414 CF7Q9W 142737965 IC50 = 159 nM T63414 C2AE5F 145949409 IC50 = 10 nM T63414 CVUB13 145951660 IC50 = 62 nM T63414 C6MJF8 145951717 IC50 = 6 nM T63414 CT3YR8 145952273 IC50 = 54 nM T63414 CLV0D9 145953487 IC50 = 85 nM T63414 C0L3XO 145953515 IC50 = 723 nM T63414 C5F8OS 145953552 IC50 = 263 nM T63414 CW1ZS3 145953795 IC50 = 621 nM T63414 CYA15N 145954765 IC50 = 434 nM T63414 CI0BL7 145954866 IC50 = 8 nM T63414 C1H3YT 145956657 IC50 = 810 nM T63414 C8N4CA 145957051 IC50 = 120 nM T63414 CUK8L0 145957428 IC50 = 335 nM T63414 CBEA20 145958746 IC50 = 10 nM T63414 CYR3O9 145959117 IC50 = 12 nM T63414 CJ5XS2 145959607 IC50 = 18 nM T63414 CXPW20 145959674 IC50 = 108 nM T63414 CLS0X7 145960885 IC50 > 10000 nM T63414 CQK90X 145961422 IC50 = 7 nM T63414 C7M1NU 145962280 IC50 = 123 nM T63414 CD9P3E 145972418 IC50 = 861 nM T63414 CVO0B7 145972899 IC50 = 888 nM T63414 C5ZPH0 145974559 IC50 = 73 nM T63414 CQH5J2 155511022 Ki = 2.5 nM T63414 CPE58H 155514125 IC50 > 15000 nM T63414 CF6LV4 155514310 IC50 > 30000 nM T63414 C8F0TD 155517593 IC50 = 19 nM T63414 C5RO9U 155518243 IC50 = 103 nM T63414 CXV48Z 155520870 IC50 = 3.6 nM T63414 C1M6UJ 155522112 IC50 = 8.5 nM T63414 C1B9FT 155522567 IC50 = 7.4 nM T63414 CF7OT4 155523772 IC50 = 230 nM T63414 CM9CW2 155526224 IC50 > 100000 nM T63414 C1NOD4 155529242 IC50 > 100000 nM T63414 CX12AU 155529713 IC50 = 8530 nM T63414 C5BC9V 155529971 IC50 > 100000 nM T63414 CH0E9W 155530155 IC50 = 3.2 nM T63414 CP83MR 155530812 IC50 = 4.5 nM T63414 COU59G 155533299 IC50 = 22 nM T63414 C9DC1A 155534002 IC50 < 10 nM T63414 CL2YH0 155539805 IC50 = 3.9 nM T63414 COD7Q8 155543044 IC50 > 100000 nM T63414 CJVB92 155551147 Ki = 1.9 nM T63414 CZ9G8K 155559078 IC50 > 100000 nM T63414 C0PYX1 155562454 IC50 > 30000 nM T63414 C06HKI 155563184 IC50 = 3.4 nM T63414 CKOT58 155566246 IC50 = 44 nM T63414 CBS9Q8 10022445 IC50 = 6.31 nM T63414 CQB54V 11497646 IC50 = 25.12 nM T63414 C3D9RS 11526539 IC50 = 15.85 nM T63414 C9KV7B 11698695 IC50 = 79.43 nM T63414 CX24BZ 11741157 IC50 = 10 nM T63414 CR7HA4 135448190 IC50 = 100 nM T63414 CPXN13 135458217 IC50 = 63.1 nM T63414 C0G7OE 135965987 IC50 = 39.81 nM T63414 CBE09L 135966074 IC50 = 125.89 nM T63414 CT9RX6 136018716 IC50 = 398.11 nM T63414 CLU32R 19796273 IC50 = 15.85 nM T63414 CS3Q5J 23725174 IC50 = 79.43 nM T63414 C93RSL 24894834 IC50 = 1 nM T63414 CJBV47 24994779 IC50 = 398.11 nM T63414 CU8FD3 25013922 IC50 = 0.3981 nM T63414 C0WH3T 2818099 IC50 = 3981.07 nM T63414 CH96RX 45267182 IC50 = 199.53 nM T63414 CE2A7D 45267983 IC50 = 0.07943 nM T63414 CB1KJ0 45268902 IC50 = 31.62 nM T63414 C90SVN 45269779 IC50 = 316.23 nM T63414 C46KDJ 45270539 IC50 = 1.259 nM T63414 C89OVT 45271362 IC50 = 15.85 nM T63414 CYFG04 45271369 IC50 = 3.162 nM T63414 CDK3Y5 45271370 IC50 = 2.512 nM T63414 C23POI 45271376 IC50 = 79.43 nM T63414 COU15N 45273183 IC50 = 199.53 nM T63414 C2DL7Y 9865961 IC50 = 3.981 nM T63414 D00QLM 91557 EC50 > 100000 nM T63414 D02TNK 16121950 IC50 = 1800 nM T63414 D05DLI 16121949 IC50 = 700 nM T63414 D05QLT 11673921 IC50 = 123.03 nM T63414 D07QYU 4881 IC50 = 1180 nM T63414 D08DOG 25130235 IC50 > 100000 nM T63414 D0B1KT 15953802 IC50 > 10000 nM T63414 D0H2MA 6324599 IC50 = 536 nM T63414 D0M0XC 53325875 IC50 = 6.607 nM T63414 D0N6ES 5312126 IC50 = 12.59 nM T63414 D0Q1PO 53325874 IC50 = 9 nM T63414 D0U5ML 23232014 IC50 = 39.81 nM T53350 C1GR4N 9828276 IC50 = 10 nM T53350 C32JRZ 9843079 IC50 = 19000 nM T53350 CSM41Q 9849291 IC50 = 93 nM T53350 C94WDV 9858438 IC50 = 23 nM T53350 C4P5GL 9868381 IC50 = 60 nM T53350 CJ8DP1 9868672 IC50 = 290 nM T53350 CX9N3C 9870477 IC50 = 410 nM T53350 CU3TI0 9873209 IC50 = 73 nM T53350 C9KUZ3 9880993 IC50 = 31 nM T53350 CCO0V9 9885413 IC50 = 4500 nM T53350 CBD1T3 9887686 IC50 = 1000 nM T53350 CD79UJ 9890632 IC50 = 7 nM T53350 C5DW9S 9902427 IC50 = 28 nM T53350 C8NP7J 9915263 IC50 = 30 nM T53350 C1P5HF 9916545 Ki = 8 nM T53350 C5QFN3 9922714 IC50 = 122 nM T53350 CN4YK1 9923900 IC50 = 17 nM T53350 CG1A6B 9924640 IC50 = 9.3 nM T53350 CC5R1I 9925298 IC50 = 24 nM T53350 CPU59E 9928357 IC50 = 3000 nM T53350 C1OUM6 9936924 IC50 = 470 nM T53350 CMI06Q 9939403 Ki = 43 nM T53350 CWZC93 9947332 IC50 = 21 nM T53350 CZA4H5 9967696 IC50 = 21 nM T53350 CH4SM7 9968401 IC50 = 19 nM T53350 C8AQV3 9968741 IC50 = 2 nM T53350 CTC47X 9968907 IC50 = 92 nM T53350 C8K5VD 9969928 IC50 = 33 nM T53350 CC9KU8 9982365 IC50 = 9600 nM T53350 CM4AL0 10001331 IC50 = 160 nM T53350 C6MXW1 10054053 Ki = 7 nM T53350 CVTD42 10078499 Ki = 100 nM T53350 CYE7V4 10109052 IC50 = 23 nM T53350 CJG06C 10109498 IC50 = 10 nM T53350 CQ95BV 10109888 IC50 = 30 nM T53350 C9FGV3 10110893 IC50 = 98 nM T53350 CY6HZ7 10111132 IC50 = 26 nM T53350 CV9CN8 10111662 IC50 = 17 nM T53350 CQ0B1I 10112489 IC50 = 15 nM T53350 CHC04U 10112623 IC50 = 21 nM T53350 CJD98F 10117482 IC50 = 17 nM T53350 C6O2CN 10132603 IC50 = 6 nM T53350 CC4W1H 10132648 IC50 = 45 nM T53350 CZM7F4 10132758 IC50 = 36 nM T53350 CG1WB8 10133038 IC50 = 25 nM T53350 CH7A1G 10133089 IC50 = 23 nM T53350 CE0TP5 10134393 IC50 = 5 nM T53350 CI83LM 10136534 IC50 = 57 nM T53350 CXVW40 10155383 IC50 = 14 nM T53350 CXR42J 10155792 IC50 = 3 nM T53350 CIU30R 10156141 IC50 = 6 nM T53350 C23GXV 10159719 IC50 = 17 nM T53350 C0XWZ7 10160466 IC50 = 88 nM T53350 CF81HQ 10179230 IC50 = 17 nM T53350 CNK76U 10179252 IC50 = 38 nM T53350 C0F6JV 10180091 IC50 = 30 nM T53350 CEWF13 10180993 IC50 = 65 nM T53350 CW9DP6 10182462 IC50 = 26 nM T53350 CDS9A3 10184459 IC50 = 33 nM T53350 CJ64WB 10204279 IC50 = 26 nM T53350 CQI6D5 10205950 IC50 = 14 nM T53350 CYS9I2 10222243 IC50 = 25 nM T53350 CPSX26 10256361 Ki = 14 nM T53350 C1LR9B 10269446 IC50 = 29 nM T53350 CIRH04 10270164 IC50 = 6 nM T53350 CBE81L 10270207 IC50 = 17 nM T53350 C7HZ1M 10270281 IC50 = 32 nM T53350 C9P6RD 10271010 IC50 = 43 nM T53350 C3XD1E 10271240 IC50 = 21 nM T53350 C2MES9 10271604 Ki = 11 nM T53350 CSMH63 10272472 IC50 = 26 nM T53350 CWJ02G 10273315 IC50 = 37 nM T53350 CA6W7R 10279808 IC50 = 1.8 nM T53350 CU6QR7 10291655 IC50 = 324 nM T53350 CJTV12 10293283 IC50 = 8 nM T53350 C1JDV9 10294045 IC50 = 13 nM T53350 C5KW8A 10297713 IC50 = 107 nM T53350 CX6GU9 10462047 IC50 = 26 nM T53350 CE7G5A 10570770 IC50 = 18000 nM T53350 CB20LM 10594000 IC50 = 16000 nM T53350 C9OIB3 10686890 IC50 = 112000 nM T53350 CR3Q8Z 10691191 IC50 = 29000 nM T53350 C2DZT7 11399358 IC50 = 380 nM T53350 CAK3T6 11857267 IC50 = 300 nM T53350 C7GMV4 15923505 IC50 = 67 nM T53350 C81HZU 16748676 IC50 = 116 nM T53350 CM9A3U 16748677 IC50 = 154 nM T53350 CIA12S 16748678 IC50 = 32 nM T53350 CHJ8F5 16748680 IC50 = 3 nM T53350 CG7PV5 16748681 IC50 = 184 nM T53350 CT9B6F 16748784 IC50 = 6 nM T53350 CY9B0N 16748785 IC50 = 14 nM T53350 CU8WG1 16748786 IC50 = 74 nM T53350 CJ5RN8 16748788 IC50 = 46 nM T53350 C6F9LM 16748789 IC50 = 6 nM T53350 C0D4MW 16748790 IC50 = 59 nM T53350 CP05WD 16748896 IC50 = 18 nM T53350 CO2Q0D 16748897 IC50 = 13 nM T53350 C5VYB0 16748898 IC50 = 28 nM T53350 CXB10H 16748901 IC50 = 6 nM T53350 CYZ7R6 16749000 IC50 = 28 nM T53350 CJ1V6K 18325275 IC50 = 34000 nM T53350 C9FH2C 18337540 IC50 = 53 nM T53350 CR7JL9 18678862 IC50 = 1700 nM T53350 CG23VF 18678893 IC50 = 42000 nM T53350 C9EL0C 18678910 IC50 = 6700 nM T53350 CCX05P 18678912 IC50 = 900 nM T53350 C0XA5P 18678938 IC50 = 9100 nM T53350 CES6T4 23553780 IC50 = 8100 nM T53350 CL5C3M 23553781 IC50 = 81000 nM T53350 CA70EU 23553786 IC50 = 1000 nM T53350 CH4LV7 44273823 IC50 = 4.6 nM T53350 C5SW2F 44273953 IC50 = 37 nM T53350 CO4YF9 44273954 IC50 = 30 nM T53350 CLB7X0 44273997 IC50 = 200 nM T53350 C8NOD4 44273998 IC50 = 32 nM T53350 CE1NZ7 44273999 IC50 = 27 nM T53350 CT46MN 44274026 IC50 = 10 nM T53350 CN3WI7 44274027 IC50 = 860 nM T53350 C9ZL8U 44274028 IC50 = 9 nM T53350 C9FDN7 44274049 IC50 = 290 nM T53350 CH0OQ4 44274050 IC50 = 610 nM T53350 CY4MW8 44274066 IC50 = 670 nM T53350 CS6DI7 44274067 IC50 = 60 nM T53350 C72GYW 44274068 IC50 = 590 nM T53350 C2RI4D 44274069 IC50 = 32 nM T53350 C1WI6L 44274070 IC50 = 3.9 nM T53350 CTZ4I5 44274085 IC50 = 180 nM T53350 CY6W3R 44274086 IC50 = 592 nM T53350 CEG7R4 44274087 IC50 = 200 nM T53350 CE8H6I 44274103 IC50 = 170 nM T53350 C0IZ1H 44274105 IC50 = 120 nM T53350 CP3QO4 44274112 IC50 = 230 nM T53350 C1ASR6 44274113 IC50 = 230 nM T53350 CK20ZL 44274114 IC50 = 490 nM T53350 C43QAO 44274115 IC50 = 26 nM T53350 CUHA75 44274116 IC50 = 14 nM T53350 C9NWA5 44274119 IC50 = 210 nM T53350 CJE3L8 44274120 IC50 = 80 nM T53350 CAR8E4 44274121 IC50 = 110 nM T53350 CT6ZL8 44274122 IC50 = 180 nM T53350 C3TU4Y 44274123 IC50 = 260 nM T53350 CM49SA 44274124 IC50 = 120 nM T53350 CX9KL8 44274125 IC50 = 60 nM T53350 CJB2P6 44274138 IC50 = 440 nM T53350 CNOR83 44274139 IC50 = 190 nM T53350 C1UJ9L 44274140 IC50 = 24 nM T53350 C9I0LH 44274141 IC50 = 440 nM T53350 CR86EB 44274143 IC50 = 45 nM T53350 C3A0SC 44274144 IC50 = 40 nM T53350 CF1J9A 44274147 IC50 = 40 nM T53350 C38ALF 44274154 IC50 = 150 nM T53350 C72XAT 44274155 IC50 = 220 nM T53350 C9M4WO 44274156 IC50 = 390 nM T53350 CXO3T1 44274172 IC50 = 18 nM T53350 CK81FD 44274173 IC50 = 16 nM T53350 C96AKO 44274203 IC50 = 110 nM T53350 C21PRN 44274204 IC50 = 360 nM T53350 C27ZDC 44274205 IC50 = 100 nM T53350 CWTA79 44274218 IC50 = 70 nM T53350 CMCU38 44274219 IC50 = 220 nM T53350 CAM42I 44274231 IC50 = 36 nM T53350 C7PQW0 44274236 IC50 = 220 nM T53350 CZ2C1V 44274249 IC50 = 24 nM T53350 C59QHS 44274259 IC50 = 0.024 nM T53350 C4AC8N 44274266 IC50 = 93 nM T53350 C2KW9H 44274279 IC50 = 23 nM T53350 CSI8T7 44274281 IC50 = 52 nM T53350 CU5HD8 44274283 IC50 = 90 nM T53350 C4YK7D 44274293 IC50 = 380 nM T53350 C08XYH 44274294 IC50 = 350 nM T53350 CH1VP7 44274296 IC50 = 80 nM T53350 CBFJ67 44274297 IC50 = 50 nM T53350 CEFC32 44274298 IC50 = 76 nM T53350 CRKY46 44274304 IC50 = 50 nM T53350 C3AQ6Z 44274305 IC50 = 470 nM T53350 C8O2UH 44274306 IC50 = 380 nM T53350 CB57JP 44274308 IC50 = 6 nM T53350 CJ4MF1 44274321 IC50 = 23 nM T53350 C4OAW3 44274325 IC50 = 280 nM T53350 C79DWQ 44274335 IC50 = 490 nM T53350 C1K6BZ 44274336 IC50 = 470 nM T53350 CY9FG8 44274337 IC50 = 28 nM T53350 C3KE8M 44274338 IC50 = 250 nM T53350 C6TS1K 44274339 IC50 = 230 nM T53350 C31AUX 44274344 IC50 = 140 nM T53350 C4WTX2 44274345 IC50 = 130 nM T53350 C5Z1BX 44274346 IC50 = 120 nM T53350 C5HT9O 44298830 Ki = 530 nM T53350 C01FXR 44305976 IC50 = 170 nM T53350 C8TCI0 44305987 IC50 = 7800 nM T53350 C80BHF 44306001 IC50 = 6900 nM T53350 C47FRM 44306006 IC50 = 5500 nM T53350 CB83EW 44306022 IC50 = 5900 nM T53350 C1QEZ4 44306024 IC50 = 4000 nM T53350 CA65HW 44306031 IC50 = 160 nM T53350 CJP86D 44306032 IC50 = 110 nM T53350 C4Z3SB 44306046 IC50 = 5000 nM T53350 CI74SL 44306059 IC50 = 160 nM T53350 C2L3DS 44306061 IC50 = 140 nM T53350 CDAO08 44306089 IC50 = 1600 nM T53350 CQ54SA 44306104 IC50 = 45 nM T53350 C04ATH 44306105 IC50 = 38 nM T53350 CL81ID 44306111 IC50 = 4500 nM T53350 CJD9F3 44306112 IC50 = 1700 nM T53350 CAK90V 44306133 IC50 = 3400 nM T53350 CS5JA7 44306166 IC50 = 990 nM T53350 C8R5ED 44306169 IC50 = 61000 nM T53350 CYQA43 44306173 IC50 = 1600 nM T53350 CQ59PY 44306174 IC50 = 1400 nM T53350 CB5DP9 44306197 IC50 = 2300 nM T53350 CYH0S5 44306198 IC50 = 120 nM T53350 CD0EC6 44306207 IC50 = 23000 nM T53350 CFP38L 44306216 IC50 = 260 nM T53350 CUQ3M0 44306231 IC50 = 2300 nM T53350 CK1AZ5 44306250 IC50 = 58 nM T53350 C59LJH 44306251 IC50 = 50 nM T53350 CCJD47 44306255 IC50 = 910 nM T53350 CT4ER7 44306282 IC50 = 230 nM T53350 CN1X5U 44306301 Ki = 840 nM T53350 CAO79R 44306320 IC50 = 50 nM T53350 C4A1NU 44306323 IC50 = 97 nM T53350 CQ73OB 44306340 IC50 = 220 nM T53350 C9JU3H 44306342 Ki = 1010 nM T53350 COA2K7 44306344 IC50 = 45 nM T53350 CJOW08 44306353 IC50 = 290 nM T53350 CKOV20 44306362 IC50 = 7200 nM T53350 CAL78Z 44306370 Ki = 530 nM T53350 C9I1FG 44306381 IC50 = 92 nM T53350 CF3N8R 44306382 IC50 = 55 nM T53350 CYGB58 44306387 Ki = 28 nM T53350 C4ZVY9 44306397 IC50 = 78 nM T53350 CRJF47 44306406 Ki = 2500 nM T53350 C5OE6X 44306446 Ki = 1960 nM T53350 CO15BI 44306454 IC50 = 970 nM T53350 CEZ4L1 44306461 Ki = 86 nM T53350 C8KLP7 44306466 IC50 = 770 nM T53350 CW76MS 44306477 IC50 = 98 nM T53350 CTF39X 44306653 IC50 = 3600 nM T53350 CTF59Q 44306688 IC50 = 2100 nM T53350 COL7D9 44306723 IC50 = 1600 nM T53350 CFR9C0 44306781 Ki = 350 nM T53350 C7WG8A 44306791 Ki = 18 nM T53350 C9IJA0 44306792 Ki = 22 nM T53350 C5AJC4 44306813 Ki = 250 nM T53350 CDSF90 44306881 Ki = 960 nM T53350 CK4X2J 44306882 Ki = 410 nM T53350 C7BQ1I 44306927 Ki = 470 nM T53350 C1O2WB 44306928 Ki = 470 nM T53350 CP5XW3 44316117 Ki = 1200 nM T53350 C3FKY0 44316219 Ki = 480 nM T53350 C80EJB 44316220 Ki = 340 nM T53350 CCR96I 44316223 Ki > 40000 nM T53350 C3KO1L 44316224 Ki = 1300 nM T53350 C9JK5P 44316233 Ki = 33 nM T53350 C9OGB4 44316243 Ki = 120 nM T53350 CG0JD3 44316269 Ki = 110 nM T53350 C29VZC 44316280 Ki = 100 nM T53350 C3LDO9 44316287 Ki = 330 nM T53350 CP4DB2 44316304 Ki = 400 nM T53350 CF68JY 44316352 Ki > 40000 nM T53350 C5JU8G 44316384 Ki = 190 nM T53350 CLPI02 44316395 Ki > 40000 nM T53350 C7DR9J 44316410 Ki = 740 nM T53350 CT2WR0 44316411 Ki = 210 nM T53350 C1O6PM 44316416 Ki = 200 nM T53350 C68WVE 44316417 Ki > 1000 nM T53350 C9BW2T 44316431 Ki = 160 nM T53350 CLE51T 44316432 Ki = 620 nM T53350 CMJ5L3 44316433 Ki > 1000 nM T53350 C4TX3K 44316457 Ki = 1000 nM T53350 CP83EX 44316470 Ki = 63 nM T53350 C6Y7JO 44316471 Ki = 105 nM T53350 CD1HN0 44316491 Ki = 11 nM T53350 CAO35N 44316499 Ki = 98 nM T53350 CP46US 44316541 Ki = 40 nM T53350 CTM97P 44316585 Ki = 35 nM T53350 CJN80M 44316602 Ki = 1170 nM T53350 CO91HP 44316604 Ki = 300 nM T53350 CO6X2Z 44316605 Ki = 410 nM T53350 C20WNF 44316625 Ki = 1200 nM T53350 C0JK1Y 44316645 Ki = 280 nM T53350 CAQ56J 44316671 Ki = 15000 nM T53350 CKXI38 44316840 Ki = 90 nM T53350 C7CDN8 44316841 Ki = 260 nM T53350 CLOS38 44316842 Ki = 64 nM T53350 C9P7CY 44316843 Ki = 340 nM T53350 CJM90I 44316904 Ki = 660 nM T53350 CFX49E 44316925 Ki = 20 nM T53350 C2W9LI 44316927 Ki = 950 nM T53350 C7B9SL 44318117 IC50 = 90 nM T53350 C3SX8W 44318148 IC50 = 3400 nM T53350 CQ6TC7 44318149 IC50 = 750 nM T53350 CG2W9I 44318150 IC50 = 3000 nM T53350 C1ED4K 44318203 IC50 = 89 nM T53350 C0EH9V 44318204 IC50 = 50 nM T53350 C32ZDF 44318243 IC50 = 53 nM T53350 C24DQK 44318245 IC50 = 18000 nM T53350 C7XUE2 44318272 IC50 = 2500 nM T53350 C7G2RX 44318273 IC50 = 94 nM T53350 CBEZ01 44318274 IC50 = 130 nM T53350 CI7C8G 44318288 IC50 = 68000 nM T53350 C2F9XO 44318296 IC50 = 22000 nM T53350 CPJ16Z 44318297 IC50 > 800000 nM T53350 CWGZ92 44318298 IC50 = 200 nM T53350 CF1C9X 44318301 IC50 = 73 nM T53350 C30HZP 44318306 IC50 = 5100 nM T53350 CXK60H 44318313 IC50 = 19000 nM T53350 CA47VD 44318314 IC50 = 67000 nM T53350 C2NZ0E 44318318 IC50 = 19000 nM T53350 CO6W8R 44318319 IC50 = 15000 nM T53350 CG82RJ 44318322 IC50 = 190 nM T53350 CQI7M0 44318329 IC50 = 3600 nM T53350 CH1Q0L 44318330 IC50 = 2100 nM T53350 C03UAX 44318331 IC50 = 20000 nM T53350 C2MV3S 44318338 IC50 = 30 nM T53350 C3GRC5 44318342 IC50 = 5000 nM T53350 CZ5C6F 44318356 IC50 = 78 nM T53350 C80SHT 44318357 IC50 = 78 nM T53350 C2FKY8 44318358 IC50 = 67 nM T53350 CGL90Q 44318414 IC50 = 43 nM T53350 CQR2A6 44318427 IC50 = 32 nM T53350 C9N8LY 44318430 IC50 = 29 nM T53350 COJ62U 44318433 IC50 = 110 nM T53350 CIW74F 44318436 IC50 = 870 nM T53350 CE49MW 44318447 IC50 = 1900 nM T53350 CB7Z1P 44318448 IC50 = 500 nM T53350 C3KQ6A 44318456 IC50 = 2800 nM T53350 CRP2K0 44318459 IC50 = 1200 nM T53350 C8H9YV 44318467 IC50 = 730 nM T53350 C2GZ9S 44318550 IC50 = 90 nM T53350 CK24SZ 44318564 IC50 = 78 nM T53350 CWX35M 44318569 IC50 = 280000 nM T53350 C0T5IF 44318571 IC50 = 150 nM T53350 CXJ70N 44318604 IC50 = 200 nM T53350 CA5UZ3 44318618 IC50 = 250 nM T53350 CC28VP 44318623 IC50 = 220 nM T53350 CREH53 44318634 IC50 = 140 nM T53350 CAMI89 44318635 IC50 = 110 nM T53350 C9B7QK 44318638 IC50 = 210 nM T53350 C1X2YB 44318641 IC50 = 200 nM T53350 C9QD7J 44318698 IC50 = 44 nM T53350 CZY65J 44318699 IC50 = 43 nM T53350 CH7P8I 44318701 IC50 = 49 nM T53350 C4I6ME 44368970 IC50 = 8765 nM T53350 CIR84S 44369104 IC50 = 820 nM T53350 CC4PA1 44425137 IC50 = 75 nM T53350 C4DU9X 44425139 IC50 = 8 nM T53350 C9PE6F 44425140 IC50 = 27 nM T53350 CXAP75 44425141 IC50 = 20 nM T53350 CU5QV9 44425142 IC50 = 3 nM T53350 CW8RY1 44425150 IC50 = 6600 nM T53350 CKO5Q0 44462281 IC50 = 61 nM T53350 CP2SR3 44462304 IC50 = 65 nM T53350 C9QKB2 44462305 IC50 = 52 nM T53350 CDPC48 44462306 IC50 = 110 nM T53350 CAK94X 44563337 IC50 = 345000 nM T53350 C70UVG 44571513 IC50 = 40 nM T53350 CNLD24 44571552 IC50 > 2000 nM T53350 C8DN4W 44571586 IC50 = 73 nM T53350 C2K4VG 44571723 IC50 = 54 nM T53350 CX73PT 59033102 IC50 = 80 nM T53350 CJBV54 71450403 IC50 = 55000 nM T53350 C2OQC8 71450455 IC50 = 2200 nM T53350 CZB83P 71450456 IC50 = 400 nM T53350 C6FC0X 71450457 IC50 > 100000 nM T53350 CF2V0Z 71450458 IC50 = 28000 nM T53350 C7QK3J 71450459 IC50 = 10000 nM T53350 CGFB90 71452285 IC50 = 4700 nM T53350 CTL67I 71452286 IC50 = 42 nM T53350 CYQZ42 71452287 IC50 = 4900 nM T53350 C8J4HD 71452288 IC50 = 1700 nM T53350 CXPE73 71452290 IC50 = 40000 nM T53350 CF8YK2 71452291 IC50 = 1500000 nM T53350 CBO3M8 71452292 IC50 = 69000 nM T53350 C1KWB9 71454082 IC50 = 2300 nM T53350 CB8X0C 71454083 IC50 = 11000 nM T53350 C5J0NE 71454084 IC50 = 42000 nM T53350 CWZ7L2 71455769 IC50 = 166000 nM T53350 CQ63LJ 71455820 IC50 = 17000 nM T53350 C8YE3R 71455821 IC50 = 350 nM T53350 C7ZQB1 71455822 IC50 = 102000 nM T53350 CCDX81 71455823 IC50 = 23000 nM T53350 C10DWM 71457610 IC50 = 1000 nM T53350 CLP8O4 71457611 IC50 = 10000 nM T53350 CU69CF 71457612 IC50 = 2800 nM T53350 CUMY70 71459448 IC50 = 780 nM T53350 C5JDA8 71459505 IC50 = 73000 nM T53350 CJ15TM 71459506 IC50 = 18000 nM T53350 CFTB42 71459507 IC50 = 67000 nM T53350 C7SB0J 71459508 IC50 = 85000 nM T53350 CTBK47 71461245 IC50 = 13000 nM T53350 CGQM98 71461246 IC50 = 14000 nM T53350 CIZD69 71461247 IC50 = 9400 nM T53350 CFO6X9 71461248 IC50 = 167000 nM T53350 C6IB1K 71462974 IC50 = 7100 nM T53350 CX85QT 73346950 IC50 = 65000 nM T53350 C61RYQ 90662998 IC50 = 17000 nM T53350 CEZ3R0 91824149 IC50 < 1 nM T53350 CQ7KI2 118225750 Ki = 0.04 nM T53350 CUZ1D6 118225779 IC50 < 1 nM T53350 C4OD0K 118225789 IC50 = 32 nM T53350 CD8PA1 118225803 Ki = 0.0068 nM T53350 C6F8QV 118225829 IC50 < 1 nM T53350 C38RXZ 118225927 IC50 = 1 nM T53350 CI10PX 118225935 IC50 < 1 nM T53350 CN04JW 118225947 IC50 = 20 nM T53350 C4XUH1 118225963 IC50 = 1 nM T53350 C6E4SR 118226041 IC50 = 8 nM T53350 CLI7B8 118226146 IC50 = 25 nM T53350 C4FVJ1 135487604 IC50 = 10 nM T53350 CL9Y5Q 135678161 IC50 = 4000 nM T53350 C3AVY9 135712681 IC50 = 39 nM T53350 CJ9B6C 145963868 IC50 = 1250 nM T53350 C42AZM 145965977 IC50 > 10000 nM T53350 C8DF3N 145967770 IC50 = 160 nM T53350 CZ2XC4 145973252 IC50 = 6300 nM T53350 CZ4SB5 145976911 IC50 = 126 nM T53350 D02DQT 44274134 IC50 = 0.2 nM T53350 D0A4TC 446504 IC50 = 3000 nM T53350 D0NP8A 10370504 IC50 = 52000 nM T53350 D0P2TS 9818682 IC50 = 26 nM T49948 CNX79K 15303 IC50 = 2200 nM T49948 CFW1B7 736887 IC50 = 34000 nM T49948 CNSQ89 1241300 IC50 = 6900 nM T49948 CD2B0L 1714745 IC50 = 16000 nM T49948 CAFX17 2049595 IC50 = 79 nM T49948 C5VPU9 2735965 IC50 = 1800 nM T49948 CTVJ79 2737248 IC50 = 3400 nM T49948 CR3W9I 2769974 IC50 = 25000 nM T49948 CMP79R 2797430 IC50 = 4500 nM T49948 CY3N9K 2802558 IC50 = 280 nM T49948 C6R0PL 2811867 IC50 = 2700 nM T49948 C31SMO 2822041 IC50 = 200000 nM T49948 CDO08E 3691620 IC50 = 9000 nM T49948 CTX1Q3 4459133 IC50 = 5900 nM T49948 CXR6C0 5715203 IC50 = 530 nM T49948 C9A2SF 10658517 IC50 = 60000 nM T49948 C0KQ5I 16109339 IC50 = 82000 nM T49948 C2OT0I 16109340 IC50 = 37000 nM T49948 CKF72E 16109341 IC50 = 650 nM T49948 C13PVF 16109342 IC50 = 500000 nM T49948 C3FJH7 16109343 IC50 = 15000 nM T49948 CQ9ZK7 16109344 IC50 = 560000 nM T49948 CM4CJ3 44418971 IC50 = 6000 nM T86646 D04JEE 4946 IC50 = 4 nM T86646 D04VMT 5253 IC50 = 7200 nM T86646 D05DVP 5717 IC50 > 10000 nM T86646 D07MOX 439260 EC50 = 2600 nM T86646 D0I8FI 3779 EC50 = 30 nM T86646 D0O6IU 6041 EC50 = 6000 nM T86646 D0V4QS 135398745 Ki > 10000 nM T86646 D01VAB 2119 IC50 = 2.3 nM T86646 D08AWI 11430856 Ki > 2000 nM T86646 D0ZG9N 132337 Ki > 10000 nM T86646 CZUI83 2769 IC50 > 10000 nM T86646 CJQE97 5581 EC50 = 31 nM T86646 C4W1LV 58505 IC50 = 7000000 nM T86646 CVD0J9 66245 IC50 = 7200 nM T86646 CMWP80 121888 EC50 > 30000 nM T86646 CNWM94 489104 IC50 = 98 nM T86646 CSA6U7 489105 IC50 = 38000 nM T86646 CX6LW0 489106 IC50 = 4.3 nM T86646 C6WKB1 489107 IC50 = 25000 nM T86646 CIY21Q 547892 EC50 = 10 nM T86646 CI1O5D 9818958 IC50 = 2350000 nM T86646 CJ8LT7 9848518 IC50 > 10000 nM T86646 CT2C6K 9870702 IC50 > 10000 nM T86646 C6CZ3G 9906777 IC50 > 10000 nM T86646 CH5D3J 9928343 IC50 > 10000 nM T86646 C0FS3J 10142284 EC50 = 77 nM T86646 C6YW1R 12780318 EC50 = 20 nM T86646 C48KGC 12780320 EC50 = 30000 nM T86646 C8KVA9 14739875 IC50 = 150 nM T86646 C8D9YJ 14739876 IC50 = 43800 nM T86646 CHB84K 14739877 IC50 = 3900 nM T86646 C4QFC6 14739878 IC50 = 2900 nM T86646 CLV97P 14739879 IC50 = 192000 nM T86646 CJG6A4 14739880 IC50 = 12400 nM T86646 C2JIW3 14739881 IC50 = 61400 nM T86646 CBF70X 14739882 IC50 = 420 nM T86646 CL0ZW5 14739883 IC50 = 227000 nM T86646 CP5MC4 14739885 IC50 = 30900 nM T86646 CQBE07 14739886 IC50 = 12200 nM T86646 CB54QK 14739887 IC50 = 360000 nM T86646 CI1L9P 14739889 IC50 = 990 nM T86646 C21QMJ 14739890 IC50 = 2900 nM T86646 C25HZI 14739891 IC50 = 25800 nM T86646 CV8D7G 14739892 IC50 = 780 nM T86646 C4RO8H 14739896 IC50 = 15800 nM T86646 CIR0Q4 14739897 IC50 = 15700 nM T86646 CAQ69K 14739898 IC50 = 109000 nM T86646 C42CAQ 14739899 IC50 = 293000 nM T86646 C3XY0A 14739900 IC50 = 8400 nM T86646 C1R5FU 14739901 IC50 = 2300 nM T86646 CBQT63 14739905 IC50 = 40 nM T86646 C8NO3D 14739906 IC50 = 270 nM T86646 CD4JZ0 14739907 IC50 = 90 nM T86646 CE5LK3 14739908 IC50 = 3600 nM T86646 C6YCF8 14739909 IC50 = 3700 nM T86646 CE0PW2 16116807 EC50 > 30000 nM T86646 C8WLU1 19386048 EC50 > 30000 nM T86646 C1FRU8 44288600 IC50 > 10000 nM T86646 CJ2M7V 44329832 IC50 = 15700 nM T86646 C7YO1T 44329840 IC50 = 300 nM T86646 CNW2Y0 44336319 EC50 = 10 nM T86646 CC3D1O 45260430 EC50 > 30000 nM T86646 C0EQ5X 45264302 EC50 > 30000 nM T86646 CDI84E 71450922 IC50 > 10000 nM T86646 C5OU1T 135409492 Ki > 10000 nM T86646 C4PM9W 135515431 Ki > 10000 nM T86646 D03TPY 9885123 IC50 > 10000 nM T86646 D05KUM 135446209 Ki > 10000 nM T39321 D04XGT 31593 IC50 > 50000 nM T39321 D05EAM 4735 IC50 > 50000 nM T39321 D06IAR 60961 IC50 = 50000 nM T39321 D0NQ5I 65710 IC50 = 700000 nM T39321 CTS9E0 4624 IC50 = 8000 nM T39321 CV24FH 10228 IC50 = 208929.61 nM T39321 CKN4M5 14180 IC50 > 500000 nM T39321 C2J0PB 15048 IC50 = 8000000 nM T39321 CJ8NF1 24405 IC50 > 5000000 nM T39321 C1NQ8E 65188 IC50 = 194984.46 nM T39321 C7LF0S 68229 IC50 = 123026.88 nM T39321 CQG8F3 87216 IC50 = 3700000 nM T39321 CS4QG5 92208 Ki = 2800000 nM T39321 CQJ96I 125347 IC50 = 3100000 nM T39321 C3DS1E 446186 IC50 = 7000 nM T39321 C1CW3K 459890 IC50 = 8000 nM T39321 C6WY7U 463722 IC50 = 1800000 nM T39321 CU8B6Q 467916 IC50 = 300 nM T39321 CFU1T3 759292 IC50 = 144543.98 nM T39321 C9S2LO 4055843 IC50 = 38904.51 nM T39321 CS4KE7 5287846 IC50 = 54954.09 nM T39321 CHGO41 5363192 IC50 = 162181.01 nM T39321 CI2YH7 9924682 IC50 = 34003000 nM T39321 C9GWT6 9975183 IC50 = 600000 nM T39321 C9VF0R 9998966 IC50 > 10000000 nM T39321 CQ9RT8 10019035 IC50 > 4000000 nM T39321 CJ69UL 10029114 IC50 = 4000 nM T39321 CX6R0T 10045055 IC50 = 2400 nM T39321 C5L0IR 10049523 IC50 = 500000 nM T39321 C7G0JC 10066396 IC50 = 600 nM T39321 CHT5G7 10072244 IC50 = 200000 nM T39321 C0S3CH 10318843 IC50 = 700000 nM T39321 CR6AK3 10319600 IC50 = 400000 nM T39321 CP39MN 10334943 IC50 > 4000000 nM T39321 C76SQA 10337187 IC50 = 16982.44 nM T39321 C0LTR7 10339188 IC50 = 700000 nM T39321 CLN9P6 10341490 IC50 = 3000000 nM T39321 C8YDI5 10343681 IC50 = 6300000 nM T39321 CX1C3D 10348211 IC50 > 50000 nM T39321 C0KQT5 10360939 IC50 > 2000000 nM T39321 CWN87M 10368295 IC50 = 16000 nM T39321 CE7VQ8 10381084 IC50 > 4000000 nM T39321 CSTB14 10386525 IC50 = 200000 nM T39321 C07HWY 10393235 IC50 = 26000 nM T39321 C45RCF 10405158 IC50 = 10000 nM T39321 CRHU08 10408674 IC50 = 9000000 nM T39321 CR72DH 10428340 IC50 > 10000000 nM T39321 C0R1KB 10429225 IC50 = 3300 nM T39321 CCEL76 10431926 IC50 > 10000000 nM T39321 C2RPH3 10445321 IC50 = 1600000 nM T39321 C9NBJ1 10450657 IC50 > 4000000 nM T39321 CU25FM 10454854 IC50 = 500000 nM T39321 CKF0N9 10469836 IC50 > 2000000 nM T39321 CC3J4G 10476477 IC50 = 150000 nM T39321 C4HPM8 10528348 IC50 = 1200000 nM T39321 C4H0PY 10549805 IC50 = 600000 nM T39321 CVKI74 10620158 IC50 = 850000 nM T39321 CB4HC6 10668788 IC50 = 650000 nM T39321 CZ4QK0 10697288 IC50 = 25000 nM T39321 C87ACT 10740715 IC50 = 250000 nM T39321 C0KDO7 10792034 IC50 = 25000 nM T39321 CCSJ93 10834615 IC50 = 360000 nM T39321 C8C0TX 10835695 IC50 = 500000 nM T39321 CH6FQ5 10839640 IC50 = 5500 nM T39321 CXG08M 10940514 IC50 = 14000 nM T39321 C40FAS 10974017 IC50 = 40000 nM T39321 C4W2YD 11028195 IC50 = 7000 nM T39321 CKTO76 11028555 IC50 = 14000 nM T39321 CZF75Y 11114718 IC50 = 45000 nM T39321 C4BSO1 11124571 IC50 = 25000 nM T39321 C8T2GN 11512859 IC50 = 5000 nM T39321 C79IKG 11731457 IC50 = 12000 nM T39321 CRE0O4 11753045 IC50 = 6000 nM T39321 CH1O5K 11813682 IC50 = 12000 nM T39321 CHD9S0 11814031 IC50 = 7000 nM T39321 CN6S5T 11966381 IC50 = 8000 nM T39321 C2K4CN 15828698 IC50 = 590 nM T39321 CAF6E1 21829325 IC50 = 346736.85 nM T39321 CKQ84Y 24178170 IC50 > 10000 nM T39321 CSYD02 24863870 IC50 = 17782.79 nM T39321 C0GF7M 44306170 IC50 = 5000 nM T39321 C4NRA2 44306171 IC50 = 10000 nM T39321 CYZ5O4 44306177 IC50 = 30000 nM T39321 C7I8MA 44309784 IC50 = 85113.8 nM T39321 CAG5V7 44309804 IC50 = 5000 nM T39321 C3SI8V 44309810 IC50 = 52480.75 nM T39321 CHPX93 44309822 IC50 = 56234.13 nM T39321 C4D6ZN 44309832 IC50 = 30902.95 nM T39321 CH96VA 44309844 IC50 = 128824.96 nM T39321 CR9T2D 44309846 IC50 = 12000 nM T39321 CTK17A 44309997 IC50 = 74131.02 nM T39321 CMD14G 44310158 IC50 = 123026.88 nM T39321 CMS3I2 44310159 IC50 = 67608.3 nM T39321 CT7H5Q 44310180 IC50 = 64565.42 nM T39321 CYU58F 44310181 IC50 = 190546.07 nM T39321 CFB13G 46874050 IC50 = 240000 nM T39321 CB2UL5 46875344 IC50 = 250000 nM T39321 C90BVF 46875585 IC50 > 2000000 nM T39321 C3BPX0 46875590 IC50 = 750000 nM T39321 CS7HV0 46875985 Ki = 4000000 nM T39321 CP6K1F 46875998 Ki = 9000 nM T39321 CL1MK0 46876011 Ki = 1500000 nM T39321 C5OQ1D 46876042 Ki = 800000 nM T39321 C2QSA5 46876048 Ki = 3300000 nM T39321 C39XRD 46876082 IC50 = 8000000 nM T39321 C7Q3GH 46876205 IC50 = 340000 nM T39321 C5TMK8 46876222 IC50 > 5400000 nM T39321 CO25UZ 73356664 IC50 = 29000 nM T39321 C0Y8AZ 90662838 IC50 = 45000 nM T39321 CQT9A5 118719207 IC50 = 60 nM T39321 C0UO7C 118753751 IC50 = 100 nM T39321 CF1J8L 122185475 IC50 = 1340 nM T39321 CXHN49 122185488 IC50 = 1410 nM T39321 CUFZ63 122185495 IC50 = 2410 nM T39321 C5U1BH 135476505 IC50 = 56234.13 nM T39321 D02JEZ 5281426 IC50 = 616595 nM T39321 D03RFA 657378 IC50 > 5000000 nM T39321 D03ZMQ 323 IC50 = 691830.97 nM T39321 D05QOR 5280460 IC50 = 257039.58 nM T77400 D05GJW 20279 IC50 > 10000 nM T77400 D05MQK 110635 IC50 > 10000 nM T77400 D0C9SY 135400189 IC50 = 3100 nM T77400 D0D1HW 135409400 IC50 = 34000 nM T77400 D0E0SW 53708 IC50 = 520000 nM T77400 D0F8RA 2153 IC50 = 210000 nM T77400 D0F9GE 3108 IC50 = 3600 nM T77400 D0NJ3V 4680 IC50 = 2300 nM T77400 D0R5RR 119182 IC50 = 3120 nM T77400 D0Y9ZE 4197 IC50 = 200000 nM T77400 D0Z7ZM 135398744 IC50 > 10000 nM T77400 D01LCC 17754438 IC50 > 10000 nM T77400 D07GHV 60143346 IC50 = 1 nM T77400 D0T5PO 5092 IC50 > 16000 nM T77400 D0X0PP 59351313 IC50 > 30000 nM T77400 D01ITP 71295652 IC50 = 6 nM T77400 D05VBJ 71295299 IC50 = 69 nM T77400 D07EUB 46200734 IC50 = 2.99 nM T77400 D09BDD 56933838 IC50 = 14 nM T77400 D0WS3T 72706254 IC50 = 7900 nM T77400 D00SPK 23665864 IC50 = 15000 nM T77400 D00YPW 135399235 IC50 = 46800 nM T77400 D02EMR 151170 IC50 > 10000 nM T77400 D07FHZ 5087 IC50 = 390000 nM T77400 D08NXX 5487281 IC50 = 20000 nM T77400 D09SFV 3973 IC50 = 40000 nM T77400 D09UMA 55918 IC50 = 500000 nM T77400 D0BK6B 3021729 IC50 = 380000 nM T77400 CVQ0G5 1348 IC50 > 100000 nM T77400 C03NGJ 1713 IC50 > 100000 nM T77400 CO2Y3R 3698 IC50 = 580000 nM T77400 CH8J2B 4977 Ki = 600000 nM T77400 CCJ8F0 5353 IC50 = 200000 nM T77400 CGA17S 127779 Ki = 122000 nM T77400 CR8H1B 149028 IC50 = 68000 nM T77400 CK4VZ8 152034 IC50 = 17000 nM T77400 C0YK8A 155806 IC50 = 212000 nM T77400 COK69D 156890 IC50 = 57000 nM T77400 CH2P8A 158961 Ki = 700000 nM T77400 CVN23X 158962 Ki = 600000 nM T77400 C78DLE 205964 IC50 = 8700 nM T77400 CKH1C0 220780 Ki = 22400 nM T77400 C51LJV 223726 Ki = 6900 nM T77400 C7YV8R 656066 IC50 = 170 nM T77400 C8JLO0 2243267 IC50 = 4100 nM T77400 CWO8I2 3041753 IC50 = 108000 nM T77400 CK12OT 3814427 IC50 > 100000 nM T77400 C7BQ1N 5492386 IC50 > 100000 nM T77400 C0C9HP 6610310 IC50 > 100000 nM T77400 CB40PM 6918356 IC50 = 1300 nM T77400 CFJ62Y 9799389 IC50 > 10000 nM T77400 CZH08Y 9802738 IC50 > 20000 nM T77400 C2NK8E 9888568 IC50 = 984 nM T77400 CO87TV 9994528 IC50 > 100000 nM T77400 CB9EY5 9995187 IC50 > 100000 nM T77400 C39LZS 9999105 IC50 > 100000 nM T77400 C4ST7G 10017729 IC50 > 100000 nM T77400 C1FJ8H 10039594 IC50 > 10000 nM T77400 C2MGJ7 10117650 IC50 = 1700 nM T77400 CG8RW2 10142576 IC50 = 950 nM T77400 CB7XJ2 10216985 IC50 = 4850 nM T77400 CZ1Y8D 10232923 IC50 > 100000 nM T77400 CWG85T 10406931 IC50 = 9000 nM T77400 CF5O8D 10446136 IC50 = 33700 nM T77400 C6PXC2 10471556 IC50 > 100000 nM T77400 C4CN0V 10508072 IC50 > 100000 nM T77400 C7Z9YF 10579873 IC50 > 100000 nM T77400 C1O4KV 10626842 IC50 > 100000 nM T77400 CE65JO 10650764 IC50 > 100000 nM T77400 C9FR7P 10674875 IC50 > 100000 nM T77400 C4T8PS 10816641 IC50 > 100000 nM T77400 C41XSK 11065470 IC50 > 10000 nM T77400 C45VZC 11438405 IC50 = 40 nM T77400 C4ZYH9 11547485 IC50 > 10000 nM T77400 CUK49V 11988837 Ki = 24000 nM T77400 CFIO49 11988967 Ki = 37000 nM T77400 C2D0NG 11989101 Ki = 39000 nM T77400 C65ABT 11989102 Ki > 100000 nM T77400 C1B4XD 11992634 IC50 > 2000 nM T77400 CPX16N 11993169 IC50 > 2000 nM T77400 CE41YR 13059432 IC50 = 190000 nM T77400 C7SPV8 13233881 IC50 = 280000 nM T77400 C75JTV 13233882 IC50 = 260000 nM T77400 C9NR8P 13233885 IC50 = 71000 nM T77400 C4AK6E 13233889 IC50 = 380000 nM T77400 CZ50CU 13887375 IC50 = 190000 nM T77400 CL9KE4 13936986 IC50 = 70000 nM T77400 CB28RL 13936987 IC50 = 30000 nM T77400 CASB70 14099426 IC50 = 480000 nM T77400 CI3J7R 14099427 IC50 = 34000 nM T77400 CQ1LY8 14099432 IC50 = 39000 nM T77400 CUS17I 14099444 IC50 = 330000 nM T77400 CP5JU9 14099446 IC50 = 170000 nM T77400 C17HNR 14099449 IC50 = 110000 nM T77400 CH4S8D 14280990 IC50 = 30000 nM T77400 CD1Q4U 14280991 IC50 = 10000 nM T77400 C03ZNU 14280992 IC50 = 50000 nM T77400 CZ9WG1 14280994 IC50 = 30000 nM T77400 CL4AF3 14280995 IC50 = 10000 nM T77400 C1MK5R 14280996 IC50 = 100000 nM T77400 CCTP04 14280998 IC50 > 100000 nM T77400 CXH95F 14280999 IC50 = 100000 nM T77400 CZ6N0W 14281000 IC50 = 40000 nM T77400 CR1G8Y 14281001 IC50 = 100000 nM T77400 CJ6VF1 14281004 IC50 > 100000 nM T77400 C9MY5X 14281006 IC50 = 5500 nM T77400 CUFJ35 14281010 IC50 = 7000 nM T77400 CQ8TE3 14281011 IC50 > 100000 nM T77400 CSEC89 14281012 IC50 = 60000 nM T77400 CU0J8E 14281015 IC50 = 100000 nM T77400 CDP92K 14281016 IC50 = 6000 nM T77400 C6FCS9 14281018 IC50 = 8000 nM T77400 CUDO17 14281023 IC50 = 60000 nM T77400 CZ19AJ 14281024 IC50 = 10000 nM T77400 CY8PC6 14281025 IC50 = 5000 nM T77400 CBT8K9 14281026 IC50 = 5000 nM T77400 C3F7MZ 14281027 IC50 > 100000 nM T77400 CQ2YL0 14281033 IC50 = 50000 nM T77400 CCO0S1 15005567 IC50 > 100000 nM T77400 CW0UP4 15005571 IC50 = 7000 nM T77400 CE0DR4 15005574 IC50 = 7000 nM T77400 CAQ7J2 15005576 IC50 = 3000 nM T77400 C5Z8QA 15005579 IC50 > 100000 nM T77400 CJ72ZA 15005584 IC50 > 100000 nM T77400 CVA9B0 15005585 IC50 = 20000 nM T77400 C7QZO0 15005594 IC50 > 100000 nM T77400 CRA5G0 15005604 IC50 = 10000 nM T77400 C0X4QW 15065159 IC50 = 60000 nM T77400 CDS3L9 15065160 IC50 = 60000 nM T77400 CJAW97 15065161 IC50 > 100000 nM T77400 C1PZ8C 18734933 IC50 > 16000 nM T77400 C3LJ4B 19003750 IC50 = 58000 nM T77400 CJ95TM 20146320 IC50 = 170000 nM T77400 CW96SI 23624262 IC50 = 1000 nM T77400 C4S6VD 23654252 IC50 > 50000 nM T77400 C9WGI4 24802717 IC50 = 239 nM T77400 C20VHK 24871823 IC50 = 4560 nM T77400 C93DZI 25147798 IC50 > 50000 nM T77400 CPC08B 25179287 IC50 > 50000 nM T77400 COB03R 25179478 IC50 > 50000 nM T77400 CS7RC9 42629350 IC50 = 32 nM T77400 C7SGR9 42629353 IC50 = 75 nM T77400 C9CE2J 42629699 IC50 = 116 nM T77400 CP9TE3 42629700 IC50 = 21.9 nM T77400 CICF39 42629702 IC50 = 38 nM T77400 CMIX45 42629822 IC50 = 9.5 nM T77400 CM3X9S 42629827 IC50 = 11 nM T77400 CQN26J 42629945 IC50 = 47 nM T77400 CRX87A 42629953 IC50 = 14 nM T77400 C6O5FX 42630062 IC50 = 37 nM T77400 CR2VK6 42630063 IC50 = 135 nM T77400 C1A4UY 42630064 IC50 = 64 nM T77400 CWT8E7 42630065 IC50 = 237 nM T77400 CTS74L 42630069 IC50 = 153 nM T77400 C3P1XN 42630071 IC50 = 70.5 nM T77400 C2O1WH 42630072 IC50 = 70 nM T77400 CGU0S3 42630073 IC50 = 21.6 nM T77400 C71ZNR 42630180 IC50 = 62 nM T77400 C9UZW3 42630188 IC50 = 22 nM T77400 CX9ZT6 42630190 IC50 = 305 nM T77400 C4RHY0 42630191 IC50 = 108 nM T77400 CT6RS9 42630192 IC50 = 92 nM T77400 CYLS05 42630193 IC50 = 66 nM T77400 C7J0PY 42630314 IC50 = 621 nM T77400 CJC7B8 42630315 IC50 = 194 nM T77400 CYZL43 42630317 IC50 = 165 nM T77400 CH42OZ 42630318 IC50 = 83 nM T77400 C7X5AH 42630437 IC50 = 30 nM T77400 C8L7XT 42630438 IC50 = 300 nM T77400 C5IVS3 42630440 IC50 = 138 nM T77400 CGV5A0 42630796 IC50 = 35.6 nM T77400 CW8OB3 44243146 Ki > 10000 nM T77400 C7NHE8 44279839 IC50 = 130000 nM T77400 CK8Y4F 44286951 IC50 > 50000 nM T77400 COBW92 44301890 IC50 = 43000 nM T77400 C8A2JP 44311854 IC50 = 89000 nM T77400 C5SBO6 44311855 IC50 = 18000 nM T77400 CQ0S7E 44386000 IC50 > 50000 nM T77400 CHDN54 44386045 IC50 = 13000 nM T77400 CBT82J 44386129 IC50 > 50000 nM T77400 CV1F8W 44386133 IC50 = 27000 nM T77400 CP37LE 44386323 IC50 = 20000 nM T77400 C69DVN 44386324 IC50 > 50000 nM T77400 CWE39G 44386327 IC50 = 14000 nM T77400 CL7OS2 44386388 IC50 = 14000 nM T77400 C2RTX1 44386433 IC50 = 44000 nM T77400 CPQC46 44386434 IC50 > 25000 nM T77400 CD8VL7 44387049 IC50 = 19000 nM T77400 CC9HR5 44387117 IC50 = 66000 nM T77400 C8ZUQ5 44411688 IC50 = 431 nM T77400 CBL2J9 45263650 IC50 = 4600 nM T77400 C0D2MN 46186792 IC50 = 4 nM T77400 CR1K5E 46198523 IC50 = 9.3 nM T77400 C58BSW 46198541 IC50 = 101.6 nM T77400 C1BIJ2 46198546 IC50 = 142 nM T77400 CC42ER 46198694 IC50 = 39.4 nM T77400 C0WRO9 46198713 IC50 = 13.2 nM T77400 CON1M4 46199019 IC50 = 14 nM T77400 C5AND7 46199167 IC50 = 28.6 nM T77400 CKX1A6 46199301 IC50 = 3.31 nM T77400 CZU0H7 46199329 IC50 = 14.4 nM T77400 CD9LN1 46199458 IC50 = 5.31 nM T77400 CXG34R 46199487 IC50 = 15.8 nM T77400 CAL85J 46199794 IC50 = 974 nM T77400 CZF5C0 46199795 IC50 = 1950 nM T77400 CI9EA4 46199799 IC50 = 2055 nM T77400 C26RJV 46200090 IC50 = 172 nM T77400 C5WND9 46200233 IC50 = 196 nM T77400 CKIC45 46200238 IC50 = 775 nM T77400 CS46AE 46200399 IC50 = 589 nM T77400 C1S3BK 46200706 IC50 = 110 nM T77400 C4P5QJ 46200709 IC50 = 103 nM T77400 CV8Y6W 46200711 IC50 = 4.37 nM T77400 CK1N4X 46200728 IC50 = 15.1 nM T77400 CH9FU8 46200877 IC50 = 3390 nM T77400 CEZ3V4 46200878 IC50 = 35.9 nM T77400 C36XLQ 46209046 IC50 > 10000 nM T77400 C2Q4YT 46209162 IC50 > 10000 nM T77400 CJOE41 46209386 IC50 > 10000 nM T77400 C5IMB2 46239424 Ki > 10000 nM T77400 CKR9P7 46239425 Ki > 10000 nM T77400 CI1F5C 46239840 Ki >= 770 nM T77400 C26XVS 46240044 Ki >= 4793 nM T77400 CE4JU7 46842025 IC50 > 10000 nM T77400 CR8JC2 46842169 IC50 > 10000 nM T77400 C3P2IN 46933992 IC50 >= 57000 nM T77400 C3R9SZ 46957534 IC50 = 490 nM T77400 C3DH7C 49821302 IC50 = 81 nM T77400 C9Q6KE 49821304 IC50 = 36 nM T77400 CE8Y6Q 49821305 IC50 = 128 nM T77400 C3TVS5 49821396 IC50 = 71 nM T77400 CHA5Z0 49821469 IC50 = 325 nM T77400 C1AYP0 49821627 IC50 = 112 nM T77400 C85AXR 49821714 IC50 = 411 nM T77400 CZS03D 50902030 Ki > 4274 nM T77400 CH2Z1E 50902289 Ki > 7100 nM T77400 C4HJL2 50902291 Ki > 7950 nM T77400 C6A1IU 50902549 Ki > 2000 nM T77400 C3Y2AV 50903255 Ki > 2000 nM T77400 CGF65A 54670110 IC50 > 30000 nM T77400 C90ZLC 54670399 IC50 > 30000 nM T77400 COHX27 56648495 IC50 = 11.6 nM T77400 C4TGL7 56648496 IC50 = 27.5 nM T77400 C43WOF 56648497 IC50 = 19.5 nM T77400 CM3OI5 56648498 IC50 = 13.1 nM T77400 CM09EW 56648583 IC50 = 29.9 nM T77400 CIT68E 56648584 IC50 = 11.5 nM T77400 C9U0JW 56648585 IC50 = 7.4 nM T77400 C8O9PD 56648586 IC50 = 108 nM T77400 C52KXF 56648587 IC50 = 5.4 nM T77400 C9NC5E 56648588 IC50 = 276 nM T77400 CSZ6J1 56648589 IC50 = 299 nM T77400 CH6C3L 56648679 IC50 = 24.6 nM T77400 CCY79V 56648680 IC50 = 30 nM T77400 CL6Q1H 56648681 IC50 = 17 nM T77400 CR0C8I 56648683 IC50 = 24 nM T77400 C15YZK 56648684 IC50 = 40.6 nM T77400 C9Z8TP 56648763 IC50 = 18.4 nM T77400 C0HX6Z 56648767 IC50 = 40 nM T77400 C85VDI 56648768 IC50 = 89 nM T77400 CNE96P 56648857 IC50 = 23 nM T77400 CX86AQ 56648859 IC50 = 13.6 nM T77400 CLV5E3 56648860 IC50 = 14.7 nM T77400 C6QG0A 56648861 IC50 = 619 nM T77400 CL8QN3 56648862 IC50 = 501 nM T77400 C16DEO 56648951 IC50 = 42 nM T77400 CPC3T4 56654131 IC50 > 10000 nM T77400 C0YD3P 56928304 IC50 > 5000 nM T77400 C8RO6A 56929788 IC50 > 1000 nM T77400 C0ZF1L 57328385 IC50 = 2100 nM T77400 C4EGB7 57392860 IC50 = 27 nM T77400 CG3DF1 57392948 Ki > 10000 nM T77400 CE36TV 57394695 Ki > 10000 nM T77400 CPA3D1 57403394 Ki > 10000 nM T77400 C4XMB6 58547809 IC50 > 30000 nM T77400 CEB3G9 58547814 IC50 = 3030 nM T77400 C08QVG 58547833 IC50 = 11700 nM T77400 CFVG67 58547863 IC50 = 29700 nM T77400 CYZA38 58548077 IC50 = 12900 nM T77400 CWX3N7 59320301 IC50 > 10000 nM T77400 C7PB1U 59321218 IC50 = 2.06 nM T77400 CS32XI 59321284 IC50 = 346.5 nM T77400 C23WQA 59321310 IC50 = 944 nM T77400 CX45HS 59321315 IC50 = 80.6 nM T77400 CZ6C9L 59321318 IC50 = 864 nM T77400 C1OHZ0 59321339 IC50 = 722 nM T77400 C0EP5I 59341847 IC50 > 10000 nM T77400 CHQ28A 59341978 IC50 > 10000 nM T77400 CJ0YB8 59351288 IC50 > 10000 nM T77400 CCA1H6 59351376 IC50 > 10000 nM T77400 C1SX6A 60149170 IC50 = 0.3 nM T77400 C0AFM6 60150358 IC50 = 30.3 nM T77400 CE0Q1S 60152740 IC50 = 3 nM T77400 CJK53Q 60152741 IC50 = 4 nM T77400 CZ7OU4 60163253 IC50 = 8.2 nM T77400 C6C8RD 66802145 IC50 = 4900 nM T77400 C2D7LR 66967770 IC50 = 3465 nM T77400 C5BE3L 67021512 IC50 = 6100 nM T77400 CA53BN 68181843 IC50 = 2.01 nM T77400 CFV5P9 68181883 IC50 = 0.58 nM T77400 CY8J3O 68181896 IC50 = 0.53 nM T77400 C5OD4I 68181996 IC50 = 0.82 nM T77400 C8JN6C 68182075 IC50 = 1.08 nM T77400 CTJ46X 68594477 IC50 = 11.8 nM T77400 CV4X6K 68595169 IC50 = 23 nM T77400 C8E0XY 68596001 IC50 = 269 nM T77400 CJ80VI 68596013 IC50 = 1500 nM T77400 CL2H4T 68596452 IC50 = 894 nM T77400 C93IHS 68596628 IC50 = 2375.5 nM T77400 CDZ01B 68596639 IC50 = 1150 nM T77400 C1CD9S 68596902 IC50 = 50.4 nM T77400 C7PCW0 68597211 IC50 = 1998 nM T77400 CGJB21 68597401 IC50 = 3420 nM T77400 CHK4S0 68597804 IC50 = 1270 nM T77400 C10TGO 68598825 IC50 = 1220 nM T77400 CHX52Y 69561043 IC50 = 38 nM T77400 CCN10Q 70662473 IC50 > 1000 nM T77400 COI2P3 70679302 IC50 > 10000 nM T77400 CM3OP8 70686796 IC50 = 95.9 nM T77400 CHBT91 70686797 IC50 = 522 nM T77400 CC43LF 71074083 IC50 > 10000 nM T77400 C4P0XT 71092344 IC50 > 30000 nM T77400 C6DAG4 71092519 IC50 > 30000 nM T77400 C6VX8J 71093641 IC50 = 17.7 nM T77400 C87NJD 71114298 IC50 = 9 nM T77400 CLU1S6 71151948 IC50 = 5.9 nM T77400 CY9ZL0 71151966 IC50 = 280 nM T77400 C34XNL 71151981 IC50 = 9.7 nM T77400 C82AUP 71152059 IC50 = 2.2 nM T77400 C0C9JX 71152125 IC50 = 6.3 nM T77400 C5VUO9 71152240 IC50 = 2.8 nM T77400 CGTE48 71152251 IC50 = 30 nM T77400 CY3RW6 71152297 IC50 = 0.38 nM T77400 CN8W4I 71153086 IC50 = 6.2 nM T77400 CDZ4U5 71153104 IC50 = 21 nM T77400 C2TEH0 71153106 IC50 = 6.5 nM T77400 C1M0EN 71153110 IC50 = 4.4 nM T77400 C0M7ZG 71153186 IC50 = 29 nM T77400 CG9C3J 71153201 IC50 = 7.1 nM T77400 CT8W1G 71153209 IC50 = 10.4 nM T77400 CUW9X3 71153218 IC50 = 1.4 nM T77400 CD6C7M 71153238 IC50 = 0.28 nM T77400 C2NV4G 71153252 IC50 = 15 nM T77400 C74BDZ 71153260 IC50 = 263 nM T77400 CIM4L0 71153268 IC50 = 12.1 nM T77400 CCY3I0 71153278 IC50 = 1.7 nM T77400 CVW5J0 71153282 IC50 = 7.7 nM T77400 CH51WI 71153284 IC50 = 28 nM T77400 CYX69F 71153287 IC50 = 123 nM T77400 C3V5ZM 71153302 IC50 = 4.8 nM T77400 C40HNF 71153309 IC50 = 0.6 nM T77400 CM9DL8 71153318 IC50 = 8.9 nM T77400 C9NRH4 71153321 IC50 = 0.47 nM T77400 C0B4QF 71153327 IC50 = 39 nM T77400 CF7C0J 71153330 IC50 = 0.42 nM T77400 C3DT6Q 71153343 IC50 = 24 nM T77400 C2PE4N 71153351 IC50 = 6.3 nM T77400 C2HGI7 71153408 IC50 = 10 nM T77400 CU8MY9 71153417 IC50 = 30.5 nM T77400 CZTL75 71153427 IC50 = 6.1 nM T77400 C9GR3L 71153436 IC50 = 2.8 nM T77400 CP2SO9 71295337 IC50 = 15 nM T77400 C7LRS9 71305062 IC50 = 45 nM T77400 CR5NQ6 71450591 IC50 > 10000 nM T77400 CGD56M 71450592 IC50 > 10000 nM T77400 CZ1YN2 71452430 IC50 > 10000 nM T77400 CI1M8Q 71452431 IC50 > 10000 nM T77400 CKD9F3 71453591 IC50 = 16800 nM T77400 CX5D2O 71454197 IC50 > 10000 nM T77400 CJV1G2 71455939 IC50 > 10000 nM T77400 C8A4ME 71457746 IC50 > 10000 nM T77400 C3VKH8 71459650 IC50 > 10000 nM T77400 CT2D6E 71461384 IC50 > 10000 nM T77400 C5WS8U 71488840 IC50 = 2 nM T77400 CT4G2Y 71488842 IC50 = 3.4 nM T77400 C5D4IR 71488864 IC50 = 1.6 nM T77400 C4ES6V 71498916 IC50 = 5 nM T77400 CS61KO 71520599 IC50 = 19 nM T77400 C9MO5E 71520601 IC50 = 20 nM T77400 CIEW64 71520602 IC50 = 15 nM T77400 CT3IN6 71520691 IC50 = 7.3 nM T77400 C1D7QX 71520692 IC50 = 12 nM T77400 C71QXS 71520693 IC50 = 24 nM T77400 C4GNJ3 71598545 IC50 > 1000 nM T77400 CR9UP6 71624530 IC50 = 102 nM T77400 C2YCS7 71624531 IC50 = 54 nM T77400 C40NTG 71624532 IC50 = 23 nM T77400 C8RDG9 71624638 IC50 = 328 nM T77400 C7LFJ0 71624639 IC50 = 93 nM T77400 C03GMI 71624640 IC50 = 44 nM T77400 CZ4KC3 71624641 IC50 = 105 nM T77400 CUWS89 71624642 IC50 = 97 nM T77400 C5NU1X 71624751 IC50 = 505 nM T77400 CPBJ05 71624752 IC50 = 483 nM T77400 CFD0X9 71624753 IC50 = 586 nM T77400 CMQ7N9 71624754 IC50 = 156 nM T77400 C4FC1W 71624755 IC50 = 46 nM T77400 CO7X9M 71624869 IC50 = 14 nM T77400 C3OTL4 71624870 IC50 = 40 nM T77400 C4WN1T 71624871 IC50 = 70 nM T77400 C2UZC5 71624872 IC50 = 36 nM T77400 CZF6X3 71624873 IC50 = 18 nM T77400 CBX7F6 71624993 IC50 = 7 nM T77400 CJ1K6H 71624994 IC50 = 6.8 nM T77400 CG9ZJ8 71624995 IC50 = 1.3 nM T77400 CFL69D 71624996 IC50 = 3.4 nM T77400 CV69IU 71624997 IC50 = 9.3 nM T77400 C16JZP 71625120 IC50 = 1.2 nM T77400 C5CQM8 71625121 IC50 = 1.4 nM T77400 C7XL9G 71625122 IC50 = 1.8 nM T77400 C2N1FS 71625123 IC50 = 2.5 nM T77400 C61ULV 71625124 IC50 = 2.5 nM T77400 C7Z5GP 71625256 IC50 = 3 nM T77400 C9HG4F 71682930 IC50 = 1.72 nM T77400 C68SDB 71719394 IC50 = 6309.57 nM T77400 CZ0G2X 72165213 IC50 > 10000 nM T77400 C7XRY6 72190879 IC50 = 0.61 nM T77400 CM0PF5 72190880 IC50 = 1.6 nM T77400 CQ3GD7 72704434 Ki = 18000 nM T77400 CBM61I 73293715 IC50 > 10000 nM T77400 CHR7D0 73334611 IC50 = 1860 nM T77400 CS5XE8 73353458 IC50 = 840 nM T77400 C56RIA 73354963 IC50 = 259 nM T77400 C9ODB8 73387740 IC50 = 1320 nM T77400 C5X6GJ 73387742 IC50 = 12900 nM T77400 CT1E6V 73387743 IC50 = 3520 nM T77400 C7D1SJ 73387744 IC50 = 5390 nM T77400 CG89ET 73387745 IC50 = 923 nM T77400 C74TSX 73425972 IC50 = 3010 nM T77400 CWX3M6 73425973 IC50 = 4890 nM T77400 CEH2R6 73425974 IC50 = 1310 nM T77400 C9JE6M 75815419 IC50 = 47.6 nM T77400 CV35TH 89880131 IC50 = 80 nM T77400 C4EWJ2 89880132 IC50 = 500 nM T77400 CB9WX4 89880134 IC50 = 19 nM T77400 CKJ6N7 90005993 IC50 = 8.9 nM T77400 C9K4MZ 90006051 IC50 = 5.8 nM T77400 CF03DW 90168772 IC50 > 20000 nM T77400 CM6J9K 90168778 IC50 > 20000 nM T77400 CGJV10 90654177 IC50 = 4.9 nM T77400 C5H3ZQ 90654182 IC50 = 3.6 nM T77400 C1JPD6 91844700 IC50 = 5900 nM T77400 CYQV05 92471958 IC50 = 590 nM T77400 C2KVP3 117948953 IC50 = 2.8 nM T77400 CSCY01 117949009 IC50 = 66 nM T77400 CR87FK 117949032 IC50 = 62 nM T77400 C1XO7G 117949037 IC50 = 4100 nM T77400 C6WJN9 117949055 IC50 = 210 nM T77400 C9AW8C 117949072 IC50 = 24 nM T77400 C1COK8 117949123 IC50 = 250 nM T77400 COWG40 117949132 IC50 = 42 nM T77400 C0K7WT 117949138 IC50 = 8.7 nM T77400 CA74NJ 117949190 IC50 = 40 nM T77400 C74VEM 117949221 IC50 = 39000 nM T77400 C95TVN 117949229 IC50 = 33 nM T77400 C5H2ZV 117949248 IC50 = 910 nM T77400 CXEW03 117949270 IC50 = 72 nM T77400 CI3YX1 117949294 IC50 = 7.2 nM T77400 CHXA98 117949376 IC50 = 65 nM T77400 CZMJ97 117949378 IC50 = 29 nM T77400 CT3V0U 117949430 IC50 = 610 nM T77400 C8TE0J 117949497 IC50 = 3.5 nM T77400 C8LRE7 117949499 IC50 = 8100 nM T77400 CNE15J 117949533 IC50 = 77 nM T77400 C7FS2Y 118470919 IC50 = 10 nM T77400 CX0UN8 118470985 IC50 = 1 nM T77400 C4S5ZK 118471014 IC50 = 52 nM T77400 CB10HL 118471019 IC50 = 2 nM T77400 CNU8X4 118471029 IC50 = 2 nM T77400 C9F4PB 118471136 IC50 = 1 nM T77400 CQN46O 118471355 IC50 = 3 nM T77400 CS2QF5 118471479 IC50 = 47 nM T77400 C70LGE 118471483 IC50 = 0.8 nM T77400 CDA5Y3 118471525 IC50 = 80 nM T77400 CX0TQ7 118471706 IC50 = 3 nM T77400 CAM28L 118471717 IC50 = 14 nM T77400 CLU3C7 118471813 IC50 = 679 nM T77400 C8BN2I 118472547 IC50 = 7 nM T77400 CYQ74R 118479645 IC50 = 8 nM T77400 C04JTM 118479706 IC50 = 62 nM T77400 CL65RB 118479752 IC50 = 23 nM T77400 CVYK24 118556943 IC50 > 50000 nM T77400 CRA46I 118713812 IC50 = 404 nM T77400 C6RHL2 118736439 IC50 = 10 nM T77400 CZ1AM2 118736440 IC50 = 310 nM T77400 CXP31F 118736441 IC50 = 150 nM T77400 C8L7TA 118736442 IC50 = 5750 nM T77400 CP9T3B 118736443 IC50 = 2450 nM T77400 CVX94D 118736444 IC50 = 54 nM T77400 CM1X8H 118736445 IC50 = 190 nM T77400 CBW84D 118737979 IC50 = 6 nM T77400 CLR07H 118737980 IC50 = 95 nM T77400 C4CJR8 118737981 IC50 = 21 nM T77400 CLV60Q 118737982 IC50 = 3 nM T77400 CRJE23 122185011 IC50 = 5895 nM T77400 CS6M9C 122193679 IC50 > 100000 nM T77400 CY5S7B 126615633 IC50 = 52 nM T77400 CU52TA 126615644 IC50 = 987 nM T77400 CVX7U9 127029185 IC50 > 50000 nM T77400 C4UR7D 127038167 IC50 > 1000 nM T77400 C4H2TJ 127038168 IC50 = 395 nM T77400 CL9JT8 127038169 IC50 = 23.9 nM T77400 CN9BH4 127038170 IC50 = 2.06 nM T77400 CO2CI9 127038507 IC50 > 1000 nM T77400 CRF5C6 127038508 IC50 = 481 nM T77400 CJPX60 127038509 IC50 = 10.9 nM T77400 C7X2VQ 127038510 IC50 > 1000 nM T77400 C26EAG 127038511 IC50 = 65.7 nM T77400 CTM9E4 127038512 IC50 = 29.2 nM T77400 C6AQ2U 127038513 IC50 = 162 nM T77400 C6HZ8P 127038725 IC50 > 1000 nM T77400 CV1FM0 127038868 IC50 = 78.6 nM T77400 CADU23 127038869 IC50 = 3.49 nM T77400 C50MRW 127040517 IC50 = 46.8 nM T77400 CAG7Y1 127040518 IC50 > 1000 nM T77400 CLY63Q 127040519 IC50 = 98.6 nM T77400 C95LEY 127041240 IC50 > 100000 nM T77400 CW38DL 127042532 IC50 > 100000 nM T77400 CN5E6F 129010130 IC50 = 66.6 nM T77400 CRP5D9 131801460 Ki = 14.3 nM T77400 C16OKU 131801461 Ki = 237 nM T77400 CACJ46 132489333 IC50 = 362 nM T77400 C2P1IU 134129996 IC50 > 100000 nM T77400 CLE03O 134130328 IC50 > 100000 nM T77400 CSN6J0 134130563 IC50 > 100000 nM T77400 C0A1CZ 134131162 IC50 > 100000 nM T77400 CKYQ83 134587660 Ki = 642 nM T77400 CF24SY 134587670 Ki = 2340 nM T77400 CD9O8V 134587672 Ki = 4.3 nM T77400 CB8HO3 134587679 Ki = 19.6 nM T77400 CYDI92 134587729 Ki = 5.49 nM T77400 C4D5TR 134823954 IC50 = 7 nM T77400 C9IJK1 135566935 IC50 = 13000 nM T77400 C9Y7NH 136017768 IC50 = 1.59 nM T77400 C8UF7G 136087052 IC50 > 50000 nM T77400 C21FVA 136180322 IC50 = 560 nM T77400 CQW7T0 136197286 IC50 > 10000 nM T77400 C8TQ7A 136217455 IC50 > 50000 nM T77400 CMN10D 136239299 IC50 = 4.7 nM T77400 C1JUS2 137243509 IC50 > 100000 nM T77400 CPS12F 137286847 Ki = 195 nM T77400 C0KM1X 137288419 IC50 = 0.3 nM T77400 CC6TN9 137288423 IC50 = 0.6 nM T77400 CY3JA9 137348670 IC50 = 389.6 nM T77400 C50ZJS 137348671 IC50 = 7.1 nM T77400 C2N9VT 137348687 IC50 = 24 nM T77400 C64CQX 137631473 IC50 = 6100 nM T77400 C81LDE 137631646 IC50 = 3.1 nM T77400 C4OH1C 137631679 IC50 = 1200 nM T77400 C5ROI3 137631895 IC50 = 19.7 nM T77400 C2T4NC 137632277 IC50 = 16000 nM T77400 CC9T7R 137632951 IC50 = 19000 nM T77400 CU1R4L 137633190 IC50 > 100000 nM T77400 C8EV7L 137633354 IC50 = 1407 nM T77400 C6MB2D 137633899 IC50 = 21000 nM T77400 C9GJU6 137634998 IC50 = 206 nM T77400 CR31YE 137635321 IC50 = 85 nM T77400 CV6O7W 137635846 IC50 = 1.12 nM T77400 C4V0NA 137636043 IC50 = 15.6 nM T77400 CC9FP8 137636612 IC50 = 566.1 nM T77400 CME0R4 137636707 IC50 = 1000 nM T77400 C5NI2X 137636797 IC50 = 2107.4 nM T77400 C9XEK5 137637921 IC50 = 1520 nM T77400 CN7V2B 137638577 IC50 = 240.8 nM T77400 C2WA0G 137639069 IC50 = 27.7 nM T77400 CYXT20 137639195 IC50 = 792 nM T77400 CT3S0X 137640086 IC50 = 0.06 nM T77400 CKZ1V3 137640292 IC50 = 188.7 nM T77400 C13LPR 137640386 IC50 = 9.35 nM T77400 CAZJ94 137640735 IC50 = 0.92 nM T77400 CHJT03 137641277 IC50 = 146.4 nM T77400 CQ9TY5 137641733 IC50 = 70.1 nM T77400 C5E6TK 137642260 IC50 > 100000 nM T77400 C2F3KD 137642905 IC50 = 7000 nM T77400 C6VLU7 137642977 IC50 = 53 nM T77400 C9U8MJ 137643050 IC50 = 6500 nM T77400 CQP09A 137643189 IC50 = 480 nM T77400 C6ZIA0 137644259 IC50 = 5.94 nM T77400 CT95ED 137644401 IC50 = 7.8 nM T77400 CEW71T 137644414 IC50 = 2.4 nM T77400 C1L2AE 137644548 IC50 > 2000 nM T77400 CWUB18 137644904 IC50 = 5323.8 nM T77400 CY4K9V 137644985 IC50 = 297.8 nM T77400 CZ39VR 137645038 IC50 = 12 nM T77400 C4HC3F 137645688 IC50 = 1.3 nM T77400 CN7A5B 137645846 IC50 = 6.42 nM T77400 CF8PN0 137646373 IC50 = 1400 nM T77400 CH5T1N 137646636 IC50 = 24.4 nM T77400 C62WDH 137646854 IC50 > 100000 nM T77400 C27HUA 137647134 IC50 = 11 nM T77400 C9ILV2 137647474 IC50 = 49000 nM T77400 CIX4F6 137647559 IC50 = 5360 nM T77400 CYWR89 137647939 IC50 = 168 nM T77400 CHC24E 137648176 IC50 = 9.7 nM T77400 CYJ5Z4 137648284 IC50 = 3.54 nM T77400 CEI81F 137649219 IC50 = 10.9 nM T77400 C7YH2X 137649656 IC50 = 473 nM T77400 CU59SP 137649740 IC50 = 0.2 nM T77400 C4ZWI2 137649791 IC50 = 23000 nM T77400 C8YRB1 137649941 IC50 = 13.4 nM T77400 CQ21ZN 137650043 IC50 = 11.2 nM T77400 CR6M5K 137650215 IC50 = 9.26 nM T77400 CE4B5S 137651190 IC50 = 1012.7 nM T77400 CDYE95 137651309 IC50 > 100000 nM T77400 C18KXR 137651569 IC50 = 21 nM T77400 C6S2TD 137651868 IC50 = 3800 nM T77400 CIZX42 137651889 IC50 = 0.16 nM T77400 C6KX8Y 137651922 IC50 = 94.6 nM T77400 C05FML 137652023 IC50 > 100000 nM T77400 CDX5B4 137652246 IC50 = 140 nM T77400 CQ96UD 137652804 IC50 = 17.3 nM T77400 CI8OV2 137652839 IC50 = 2200 nM T77400 CIH38D 137652868 IC50 > 2000 nM T77400 CU8I3W 137653151 IC50 > 100000 nM T77400 CHLZ86 137653186 IC50 = 1.02 nM T77400 CS32XC 137653345 IC50 > 100000 nM T77400 CC5AK4 137654176 IC50 = 70000 nM T77400 CZV0W6 137654301 IC50 = 186 nM T77400 CSY3H9 137654828 IC50 = 3.59 nM T77400 CJT90A 137655626 IC50 = 423 nM T77400 CFW48A 137655833 IC50 = 0.23 nM T77400 C3EYO9 137656154 IC50 = 18.6 nM T77400 CM90RE 137656421 IC50 = 210 nM T77400 C0U1AS 137657330 IC50 = 69.2 nM T77400 CSX23V 137657865 IC50 = 28.6 nM T77400 CWC84D 137658255 IC50 = 52000 nM T77400 CM4CT5 137658915 IC50 = 199 nM T77400 CDE80H 137659658 IC50 = 3.19 nM T77400 C7FTC0 137660031 IC50 = 108.5 nM T77400 CY0V1N 137660078 IC50 = 7.8 nM T77400 C0GE7X 137660089 IC50 = 28000 nM T77400 CWAI46 137660568 IC50 = 3600 nM T77400 CTR5L7 137660971 IC50 = 28 nM T77400 C15IFJ 137662070 IC50 = 115 nM T77400 CJZD19 137662081 IC50 = 72 nM T77400 C6KYD7 137700754 IC50 > 10000 nM T77400 CM3UF7 137700779 IC50 > 20000 nM T77400 CPTE92 138319693 IC50 = 106 nM T77400 C2QLX3 138393292 IC50 > 50000 nM T77400 CSOF52 141737655 IC50 > 20000 nM T77400 C7SRA2 141737657 IC50 > 20000 nM T77400 CMIY07 141737666 IC50 > 20000 nM T77400 CC61SD 141737667 IC50 > 20000 nM T77400 C14CZJ 141737668 IC50 > 20000 nM T77400 CTNG49 141737674 IC50 > 20000 nM T77400 CJ38IC 141737676 IC50 > 20000 nM T77400 C1MC5Z 141737681 IC50 > 20000 nM T77400 CTUL23 141737690 IC50 > 20000 nM T77400 CMW20N 141737696 IC50 > 20000 nM T77400 CO1C4S 141737703 IC50 > 20000 nM T77400 CX9N1P 141737704 IC50 > 20000 nM T77400 C8HEG7 141737705 IC50 > 20000 nM T77400 CZTB36 145951354 IC50 = 6.9 nM T77400 C2AC1L 145963756 IC50 = 740 nM T77400 C2DKE6 145963778 IC50 > 10000 nM T77400 C8A3ES 145963852 IC50 > 10000 nM T77400 C6F8RD 145964089 Ki = 152 nM T77400 CN7EX8 145964626 Ki = 7810 nM T77400 CY69NH 145966741 IC50 = 620 nM T77400 C5RXC3 145967733 IC50 > 278000 nM T77400 CT89WH 145968235 IC50 = 670 nM T77400 CQ3RK6 145968854 IC50 = 233 nM T77400 CU2C0Y 145968972 IC50 = 18 nM T77400 C1U3IV 145969007 IC50 = 41 nM T77400 C7XA0G 145969034 IC50 = 66879 nM T77400 CH0ZK3 145969205 IC50 = 61 nM T77400 C8GDY6 145969532 IC50 = 1548 nM T77400 CH9I4O 145969561 IC50 = 2801 nM T77400 C2H9AP 145969697 IC50 = 422 nM T77400 CQ06JZ 145969912 IC50 = 6526 nM T77400 CP6QG9 145970031 IC50 = 5 nM T77400 CT3M9L 145971792 Ki = 11700 nM T77400 CHV59D 145971849 IC50 = 320 nM T77400 CH4D9S 145973243 IC50 = 1150 nM T77400 CCZ4U3 145974166 Ki = 97.2 nM T77400 CC7HN2 145974174 IC50 > 100000 nM T77400 C8P4GA 145974760 IC50 = 370 nM T77400 C6X3RQ 145975041 Ki = 15000 nM T77400 CWI73B 145976466 IC50 = 2.3 nM T77400 C9WR0G 145976954 Ki = 10100 nM T77400 C5N8AL 145977167 IC50 = 470 nM T77400 CUJZ04 145978143 IC50 > 10000 nM T77400 CK1BR0 145978345 IC50 > 100000 nM T77400 CVQ8I6 145978600 IC50 = 410 nM T77400 CKX3M5 145979083 IC50 = 1 nM T77400 C42ZAX 145979658 IC50 = 7.943 nM T77400 C93QTK 145979709 IC50 = 3.162 nM T77400 CA29ZL 145982452 IC50 = 3.981 nM T77400 CG7BR1 145987034 IC50 = 31 nM T77400 C5JXF1 145987164 IC50 = 1.995 nM T77400 CVMH95 145989382 IC50 = 3.162 nM T77400 CB5G0W 145990322 IC50 = 31.62 nM T77400 C0VQ7L 145990946 IC50 = 10 nM T77400 CZ6Y5L 145991256 IC50 = 5.012 nM T77400 CAM7X5 145991475 IC50 = 1.585 nM T77400 CHJ79V 145997874 IC50 > 10000 nM T77400 CM7TX2 148279038 IC50 > 100000 nM T77400 CM7N0S 155512334 IC50 = 1240 nM T77400 C9NVT8 155516688 IC50 = 3990 nM T77400 C5N0YD 155518781 IC50 = 11020 nM T77400 C7Z3CN 155520280 IC50 = 1940 nM T77400 CL8CU6 155521936 IC50 > 200000 nM T77400 CZPE14 155523280 IC50 = 5460 nM T77400 CWYF14 155523446 IC50 = 310 nM T77400 C1IJ5O 155526364 IC50 = 570 nM T77400 CC90XN 155526873 IC50 = 2630 nM T77400 CQ0AE6 155529518 IC50 = 40350 nM T77400 CT85RG 155530589 IC50 > 200000 nM T77400 CWKJ47 155532592 IC50 = 7270 nM T77400 CG0EC3 155536215 IC50 = 5940 nM T77400 CI4P1H 155537948 IC50 > 50000 nM T77400 C9J6VO 155540253 IC50 = 4280 nM T77400 CJ4GX7 155541617 IC50 = 3910 nM T77400 CMI8D9 155547380 IC50 = 4320 nM T77400 CSI4V9 155549683 IC50 = 5800 nM T77400 CX8DM0 155559762 IC50 = 16980 nM T77400 C9DMS4 155560624 IC50 > 50000 nM T77400 C2DA1W 155561694 IC50 = 72 nM T77400 C27FUB 155564688 IC50 = 3790 nM T77400 CQ2R0W 155568588 IC50 = 81 nM T77400 CWF2G3 71153391 IC50 = 1 nM T77400 D00YPO 14032753 IC50 = 46000 nM T77400 D05HFD 13936971 IC50 > 100000 nM T77400 D09GTN 13936969 IC50 > 100000 nM T77400 D09RKU 46239428 Ki > 10000 nM T77400 D0C2UJ 8974 IC50 > 10000 nM T77400 D0I6XA 149784 IC50 = 800 nM T77400 D0KD6S 44278378 IC50 = 17000 nM T77400 D0N6MR 10867033 IC50 = 80000 nM T77400 D0NI4Z 13936972 IC50 > 100000 nM T77400 D0R6MT 3758 IC50 = 4000 nM T77400 D0RC4F 72103 IC50 = 80000 nM T77400 D0T3UP 13724742 IC50 > 100000 nM T77400 D0V4WB 149790 IC50 = 635 nM T77400 D0V9MI 135564787 IC50 = 0.03 nM T77400 D0W3RR 10359339 IC50 = 6000 nM T07400 C9YJR2 9810788 IC50 < 500 nM T07400 CCO4K2 10188384 IC50 = 1750 nM T07400 C9WH7Y 24752728 Ki = 25 nM T07400 CL4VY2 71452357 IC50 = 1140 nM T07400 CLRZ53 71452359 IC50 = 5590 nM T07400 CE6QZ1 71452360 IC50 = 1240 nM T07400 CG1NU6 71452361 IC50 = 910 nM T07400 C6AYO7 71453726 IC50 = 16500 nM T07400 CFZ02E 71454135 IC50 = 1580 nM T07400 COE1Q3 71454136 IC50 = 1120 nM T07400 CCR73G 71455466 IC50 = 4600 nM T07400 C2D6WB 71455869 IC50 = 1210 nM T07400 C8M3TK 71455870 IC50 = 1910 nM T07400 CS8R7U 71455871 IC50 = 1720 nM T07400 CBP13J 71457675 IC50 = 1040 nM T07400 C27DBE 71457676 IC50 = 3180 nM T07400 CV9AI4 71459573 IC50 = 660 nM T07400 CI9U3N 71461319 IC50 = 1840 nM T07400 C4OH7I 71463041 IC50 = 2010 nM T07400 C6LQ4O 86304220 IC50 = 5400 nM T07400 CW1CK4 86304221 IC50 = 2500 nM T07400 CFMH38 86765239 IC50 = 1900 nM T07400 CVC9E4 86765240 IC50 = 1900 nM T07400 CGYJ35 90654926 IC50 = 18900 nM T07400 C31PFC 90654927 IC50 = 7800 nM T07400 CE0SJ3 90654928 IC50 = 5300 nM T07400 CUAO54 90664979 IC50 = 550 nM T07400 C4PN7Z 137635310 IC50 < 500 nM T40016 D04DJN 10635 IC50 = 540 nM T40016 D07BSQ 5994 Ki = 30.5 nM T40016 D0D1SG 5755 Ki = 1.14 nM T40016 D0D4HN 10607 IC50 = 14 nM T40016 D0EP0C 5833 Ki = 32.6 nM T40016 D0G3SH 31401 EC50 = 298700 nM T40016 D0G8BV 6450278 Ki = 252 nM T40016 D0IT2G 5743 EC50 = 0.1 nM T40016 D0Q4SD 443872 Ki = 3162.28 nM T40016 D0V9BD 2375 Ki > 100000 nM T40016 D0Y7IU 5281004 Ki = 1.3 nM T40016 D0Y7JU 9854489 IC50 = 0.03981 nM T40016 D0Z4EI 55245 IC50 = 0.008 nM T40016 D00JFE 56941241 IC50 = 990 nM T40016 D01SYU 10026128 IC50 = 10000 nM T40016 D03WNG 73051463 Ki = 7.2 nM T40016 D07MON 5311505 IC50 = 27 nM T40016 D07UIS 118092367 Ki = 12 nM T40016 D0HE7C 134415769 IC50 = 5.6 nM T40016 D0LI1C 44469321 IC50 > 30000 nM T40016 D0SZ1G 121248172 IC50 = 3.8 nM T40016 D0W8OJ 9854142 IC50 = 1.2 nM T40016 D0X1OW 86287635 IC50 = 9200 nM T40016 D0X9YP 67041274 IC50 = 0.056 nM T40016 D0TH6M 25204767 EC50 > 10000 nM T40016 D00PDG 44454750 Ki = 0.9 nM T40016 D02KAU 46871935 IC50 > 10000 nM T40016 D03KTE 16750192 Ki = 8300 nM T40016 D07EBU 135565424 IC50 > 10000 nM T40016 D09UFV 24825740 IC50 = 0.049 nM T40016 D0W5RL 9577221 IC50 = 120 nM T40016 C59UQE 6279 EC50 = 10 nM T40016 CD4XK3 156517 IC50 = 27000 nM T40016 CRL43B 192254 EC50 = 105300 nM T40016 CW90BT 441336 Ki = 0.7 nM T40016 C40YBS 444036 IC50 = 0.04 nM T40016 C2B0JA 674359 Ki = 1.3 nM T40016 C93EKR 674360 Ki = 26.2 nM T40016 CS6J4Z 1043068 IC50 > 100000 nM T40016 CJ02TD 3309795 IC50 > 10000 nM T40016 CKF71B 3463734 IC50 = 5700 nM T40016 CLBV35 3699263 IC50 = 480 nM T40016 C7X9AN 3728357 IC50 = 6900 nM T40016 CES83X 3775934 IC50 = 1600 nM T40016 C2EIT3 3789969 IC50 = 1300 nM T40016 C43BVE 3816305 IC50 = 735 nM T40016 CBIA94 3829166 IC50 > 10000 nM T40016 CMG30I 3832779 IC50 = 2600 nM T40016 CGH2L3 3854781 IC50 = 1800 nM T40016 CF2H8R 3865491 IC50 = 4600 nM T40016 CMK3N0 4110968 IC50 > 2000 nM T40016 C6JCL9 4163889 Ki = 33 nM T40016 C8V3MU 4193542 Ki = 24 nM T40016 CBFW65 4254945 Ki = 2.9 nM T40016 C9JP7D 4290639 Ki = 4500 nM T40016 CW23GV 4390931 Ki = 16 nM T40016 C5NDK3 4583408 IC50 > 10000 nM T40016 C0FRN6 4686093 IC50 = 4100 nM T40016 C9D6JM 4983635 IC50 > 10000 nM T40016 CBW8O6 5006871 IC50 = 2100 nM T40016 C7VQS6 5146911 IC50 > 10000 nM T40016 CDCK27 5185174 IC50 = 750 nM T40016 C16ZSG 6439929 Ki = 224 nM T40016 CG1U6P 7275458 IC50 = 55 nM T40016 CYI7T4 9802231 IC50 = 2.8 nM T40016 C7REX1 9805004 EC50 = 12.59 nM T40016 C82TUJ 9808265 IC50 = 19 nM T40016 CV87EA 9820084 IC50 = 40 nM T40016 C8A3WG 9820510 Ki > 10000 nM T40016 C06RXB 9821393 Ki = 2.1 nM T40016 C7HGB0 9822150 Ki = 236 nM T40016 CD9S5P 9825465 EC50 = 4 nM T40016 CT6OZ1 9825650 IC50 = 5.1 nM T40016 CW8LT0 9826255 IC50 = 18 nM T40016 CBS8M2 9839134 IC50 = 1756 nM T40016 C92CPK 9841404 Ki = 9200 nM T40016 CK7UC3 9841413 Ki > 10000 nM T40016 C7P6XH 9842832 Ki = 6500 nM T40016 CE9A6G 9845022 Ki = 210 nM T40016 C7RS9U 9846657 Ki = 3.3 nM T40016 CERF28 9861044 Ki = 8100 nM T40016 C3K4EU 9862027 Ki > 10000 nM T40016 CJN78I 9862597 IC50 = 35 nM T40016 C7XY1N 9863751 IC50 = 38 nM T40016 C01ZFV 9882789 IC50 = 35 nM T40016 CEM27C 9885473 Ki = 299 nM T40016 C8XSO2 9887578 Ki = 133 nM T40016 C6B9CZ 9888873 EC50 = 205 nM T40016 CZ5R9B 9890023 Ki = 11 nM T40016 CI4UK6 9890642 Ki = 2 nM T40016 CCM30W 9901180 Ki = 208 nM T40016 CJ7U3R 9904286 IC50 > 10000 nM T40016 C4KY8S 9904429 IC50 = 1316 nM T40016 C6SWK1 9904610 IC50 = 2581 nM T40016 CTI1J8 9905296 Ki = 8800 nM T40016 CE1TK2 9908041 Ki = 180 nM T40016 CG0B9U 9911589 IC50 = 3 nM T40016 CR4H6B 9919949 EC50 = 910 nM T40016 CMJG42 9921530 IC50 > 10000 nM T40016 C49UGC 9925244 Ki = 3.7 nM T40016 CUK3E9 9933829 IC50 = 26 nM T40016 C39EXP 9933936 IC50 = 430 nM T40016 CWX17A 9933946 IC50 = 707.95 nM T40016 C24FUO 9943699 IC50 = 1856 nM T40016 CXM67A 9946466 Ki = 106 nM T40016 C63MQU 9947042 Ki = 65 nM T40016 CCSX75 9949772 Ki = 1766 nM T40016 C6ZT3M 9950357 IC50 = 360 nM T40016 CKU64T 9952569 IC50 = 1 nM T40016 CW0ED9 9953456 IC50 = 146 nM T40016 CEM8L7 9969737 Ki = 2.1 nM T40016 C0Y1RE 9969849 Ki = 12.1 nM T40016 C95CAN 9978625 Ki = 0.146 nM T40016 CP2E8A 9979395 Ki = 2465 nM T40016 CP7F1R 9980041 IC50 = 7.6 nM T40016 C1QP8T 9993897 IC50 = 2500 nM T40016 COA3P9 9997031 IC50 > 2000 nM T40016 C47RUV 9998207 IC50 > 2000 nM T40016 C4V6RF 9998996 IC50 = 1.1 nM T40016 CU1ON0 9999068 Ki = 0.58 nM T40016 CL8V1C 9999671 IC50 = 565 nM T40016 CU4L7C 9999672 IC50 > 2000 nM T40016 C08OBS 10001663 IC50 > 2000 nM T40016 C0XDE9 10001914 IC50 = 194 nM T40016 CA5C6V 10002879 IC50 = 64 nM T40016 CW6P3G 10002931 IC50 = 6.3 nM T40016 C7FC9H 10004421 IC50 = 3.162 nM T40016 C3IE9K 10021634 IC50 = 355 nM T40016 CJ0O2X 10021826 IC50 > 2000 nM T40016 C52ADB 10023861 Ki = 4728 nM T40016 CN8BH3 10024007 IC50 = 5.8 nM T40016 CC4WY6 10024990 IC50 = 990 nM T40016 CSM0W3 10026120 IC50 = 690 nM T40016 C9RU8E 10027430 IC50 = 15.85 nM T40016 C9DH4U 10044332 IC50 = 0.6 nM T40016 C3ITG8 10044396 IC50 > 2000 nM T40016 C7WR0E 10044812 IC50 > 2000 nM T40016 CY6EH9 10046547 IC50 > 2000 nM T40016 C9I4JM 10046548 IC50 > 2000 nM T40016 CTL09O 10046928 EC50 = 2.7 nM T40016 CK50XF 10048063 IC50 > 2000 nM T40016 C3AXU8 10048339 EC50 = 10 nM T40016 C5E9SY 10064248 IC50 = 1.5 nM T40016 CC9Q5R 10067481 IC50 = 72.5 nM T40016 C0MG6I 10067556 IC50 > 2000 nM T40016 C2V9BW 10068183 IC50 = 710 nM T40016 CB5OZ0 10070722 IC50 = 400 nM T40016 CFY67M 10070808 Ki = 44 nM T40016 C7JQM6 10070842 IC50 = 800 nM T40016 CS9CO3 10071426 IC50 = 570 nM T40016 C9T4HR 10071810 IC50 = 77 nM T40016 C5MR6U 10071910 IC50 > 2000 nM T40016 CLO7H6 10072320 IC50 = 275 nM T40016 CUSC84 10090072 IC50 = 820 nM T40016 CQ3LD1 10091351 IC50 = 240 nM T40016 C2C7NE 10091387 IC50 > 2000 nM T40016 CRP4A3 10091735 IC50 > 2000 nM T40016 CT2Y1J 10092463 IC50 = 19 nM T40016 C16HAK 10094808 IC50 = 67 nM T40016 CC59OU 10110007 IC50 = 21 nM T40016 C3G2XJ 10110771 IC50 = 43 nM T40016 C5HM2D 10111302 IC50 = 62 nM T40016 CWR57A 10113229 Ki = 4.1 nM T40016 C62CGR 10125859 Ki = 14 nM T40016 CM4DK2 10125966 Ki = 2.7 nM T40016 CDBJ41 10126018 Ki = 9 nM T40016 CO97CW 10126196 Ki = 9.5 nM T40016 CR0DX5 10126475 IC50 = 855 nM T40016 CHS18G 10126476 IC50 = 945 nM T40016 CR0BP6 10126871 IC50 = 6.6 nM T40016 CV5PQ0 10126940 IC50 = 22 nM T40016 CVF40M 10127159 IC50 = 30 nM T40016 C3CRZ1 10127269 IC50 = 64 nM T40016 CPB60D 10127340 IC50 = 60 nM T40016 C1K8UF 10127593 IC50 = 7 nM T40016 C8VBQ0 10127709 IC50 = 9 nM T40016 CKMW98 10128037 EC50 = 45 nM T40016 C7CNX6 10128352 IC50 = 740 nM T40016 C8QRY9 10131608 IC50 = 382 nM T40016 CX6BP9 10134499 IC50 = 460 nM T40016 CWKL91 10136854 IC50 = 9 nM T40016 CS8I2Z 10138737 IC50 = 18 nM T40016 C1GI3D 10150743 IC50 = 55 nM T40016 CZKF71 10150825 IC50 = 10 nM T40016 CYR0U5 10150851 IC50 = 550 nM T40016 CVO1F7 10151165 IC50 = 24 nM T40016 C6EC1P 10151186 IC50 = 104 nM T40016 CQ14RM 10151357 IC50 = 45 nM T40016 C6U0FQ 10151473 IC50 = 61 nM T40016 CW4Y2K 10151995 IC50 = 120 nM T40016 CDV0H3 10152035 IC50 = 110 nM T40016 CR6N7C 10156793 Ki = 2.2 nM T40016 CP1M6Q 10157287 Ki = 487 nM T40016 C0MX7K 10157532 IC50 = 81 nM T40016 CKY6J8 10158491 IC50 = 41 nM T40016 CXO53S 10160645 IC50 = 28 nM T40016 C7DC1F 10162430 IC50 = 63 nM T40016 C4N8AV 10163106 IC50 = 13 nM T40016 C83WDN 10167930 IC50 = 2.1 nM T40016 CL0U4N 10172897 IC50 = 81 nM T40016 C56RYS 10173217 IC50 = 460 nM T40016 CG0VH8 10173354 IC50 = 66 nM T40016 CU6D8W 10173525 EC50 = 140 nM T40016 CP4Y6T 10173634 IC50 = 57 nM T40016 C14HMT 10173659 IC50 = 120 nM T40016 CE29WD 10174141 IC50 = 52 nM T40016 C5QDA4 10177869 IC50 = 180 nM T40016 C2P4IY 10177943 IC50 = 1430 nM T40016 CKGZ56 10178295 IC50 = 630 nM T40016 C8L7HJ 10179031 IC50 = 3 nM T40016 CNRZ84 10180123 IC50 = 10 nM T40016 CZ2L3V 10189211 IC50 = 19 nM T40016 CHK2V6 10193599 Ki = 5 nM T40016 C5SRU4 10193967 Ki = 62 nM T40016 C41YRZ 10194268 IC50 = 1125 nM T40016 CX4F7Z 10194607 IC50 = 275 nM T40016 CV0LE4 10194889 IC50 = 25.12 nM T40016 CJ1GX6 10195783 IC50 = 470 nM T40016 CRIH90 10210815 IC50 = 4.8 nM T40016 C8HDU9 10215137 EC50 = 15 nM T40016 C3O7WH 10215978 IC50 = 370 nM T40016 CX6FD1 10216117 Ki = 8.1 nM T40016 C1SG4N 10216152 IC50 = 1250 nM T40016 CD0YT7 10216465 IC50 = 46 nM T40016 C1FGX9 10216535 IC50 = 6 nM T40016 CW7QX2 10216536 IC50 = 38 nM T40016 CG9OH4 10216697 IC50 = 58 nM T40016 CXN4W1 10216788 IC50 = 580 nM T40016 CUGN98 10217411 IC50 = 77 nM T40016 C3XK0O 10217420 IC50 = 48 nM T40016 C54HJB 10221941 Ki = 9.9 nM T40016 CJ9BE0 10222329 IC50 = 7 nM T40016 CVAJ29 10223284 IC50 = 23 nM T40016 C84SRT 10223610 IC50 = 3 nM T40016 CEX46C 10224296 IC50 = 110 nM T40016 C0K1EX 10233467 IC50 = 2.2 nM T40016 CUYO17 10237223 IC50 = 610 nM T40016 C4KF2V 10237539 Ki = 511 nM T40016 CWYK62 10238100 IC50 = 15 nM T40016 C1R8GY 10238297 IC50 = 76 nM T40016 CNB1V3 10238624 EC50 = 420 nM T40016 CPGF94 10238831 IC50 = 191 nM T40016 C2AZH1 10238961 EC50 = 760 nM T40016 C56PQZ 10247253 IC50 = 116 nM T40016 CSA4R3 10252455 IC50 = 220 nM T40016 C7EGH2 10252527 IC50 = 10 nM T40016 C3C1OQ 10255490 IC50 = 3.09 nM T40016 C2N0XF 10269831 IC50 = 160 nM T40016 CR59SC 10271193 IC50 = 19 nM T40016 CPIS57 10271557 IC50 = 66 nM T40016 C4AS5M 10272127 IC50 = 216 nM T40016 CC4WT8 10272405 Ki = 13.9 nM T40016 C9UL4O 10272529 Ki = 12 nM T40016 C0D1BI 10274504 IC50 = 656 nM T40016 CKTL36 10275888 IC50 = 61 nM T40016 CQ6UW3 10283096 IC50 = 670 nM T40016 CZP75A 10286964 Ki = 8.1 nM T40016 CUQC81 10287415 IC50 > 1000 nM T40016 C5RC7X 10287444 IC50 = 30 nM T40016 CJT2G8 10287863 IC50 = 120 nM T40016 C1M6WY 10288006 IC50 = 17 nM T40016 CO6UP3 10288155 IC50 = 68 nM T40016 CNT3V9 10288528 IC50 > 2000 nM T40016 C6C2IK 10288565 IC50 = 81 nM T40016 C1I9JX 10288784 IC50 = 52 nM T40016 CNEO49 10289020 EC50 = 130 nM T40016 CMED59 10291237 IC50 = 117 nM T40016 CD03TA 10294824 IC50 = 289 nM T40016 C6TP2B 10295095 IC50 = 6 nM T40016 CZF4S5 10295116 IC50 = 9.2 nM T40016 C6JF1S 10296963 IC50 = 548 nM T40016 CUK42D 10297219 IC50 = 137 nM T40016 CLJU03 10298892 Ki = 2.4 nM T40016 C9UYG8 10309447 IC50 = 580 nM T40016 C8FM2D 10309755 IC50 = 340 nM T40016 C1OV7M 10309756 IC50 = 101 nM T40016 C9TI4A 10310063 IC50 = 56 nM T40016 CP9AE0 10310476 IC50 = 205 nM T40016 CV52EN 10310809 EC50 = 130 nM T40016 CR1L5N 10311251 EC50 = 120 nM T40016 C9FCQ5 10313926 IC50 = 194 nM T40016 C7RLW3 10314903 IC50 > 2000 nM T40016 CX7WS4 10316069 Ki = 154 nM T40016 CR9ON2 10316670 IC50 = 210 nM T40016 CP7CF8 10317646 EC50 = 21 nM T40016 CZFY94 10318044 IC50 = 804 nM T40016 CJB8R4 10319017 Ki = 331 nM T40016 CC4NU9 10319739 EC50 = 11.4 nM T40016 C7TQY8 10321412 IC50 > 2000 nM T40016 C0EJH9 10323216 IC50 = 4.677 nM T40016 C9L1FM 10325323 IC50 = 6.6 nM T40016 C6OI7M 10336208 IC50 > 2000 nM T40016 CEB82Z 10337245 Ki = 1777 nM T40016 C4QY5H 10337273 IC50 > 2000 nM T40016 C3PHW5 10339694 IC50 = 548 nM T40016 C8IAJ7 10339824 IC50 > 2000 nM T40016 CK20PF 10339825 IC50 > 2000 nM T40016 CQP1Y7 10340204 Ki = 152 nM T40016 C28SWP 10341012 IC50 > 2000 nM T40016 CQ01DG 10342379 IC50 = 980 nM T40016 CEW79S 10361500 IC50 > 2000 nM T40016 C3YU5D 10361560 IC50 = 12 nM T40016 CA20SQ 10362131 IC50 > 2000 nM T40016 CF2W3R 10362274 EC50 = 2.7 nM T40016 C2PSC1 10362449 IC50 > 2000 nM T40016 CMSA84 10362453 IC50 = 703 nM T40016 CEJ78I 10365592 IC50 = 45 nM T40016 C6QR5M 10366372 IC50 = 290 nM T40016 CDBZ06 10372181 IC50 = 86 nM T40016 C14AIB 10384345 IC50 = 34 nM T40016 C8KO5Z 10384804 IC50 = 65 nM T40016 C6RQK1 10386584 IC50 = 3.3 nM T40016 C59VXD 10386752 Ki = 0.8 nM T40016 C2MIC7 10388043 IC50 = 195 nM T40016 CBU68V 10406413 Ki = 0.95 nM T40016 C5SB4L 10407417 EC50 = 2.1 nM T40016 CEQW13 10407564 IC50 > 2000 nM T40016 CS5XF8 10408522 IC50 > 2000 nM T40016 CYZ5B6 10410448 EC50 = 5 nM T40016 C8ERB7 10411364 IC50 = 185 nM T40016 C4R6IF 10414489 IC50 = 25.12 nM T40016 CZ5CJ3 10423330 Ki = 5424 nM T40016 C3LF9D 10428026 IC50 > 2000 nM T40016 CFVP19 10428095 EC50 = 9.3 nM T40016 CJ6T4F 10428171 IC50 = 1015 nM T40016 CHR4W7 10429332 IC50 = 129 nM T40016 C03JBL 10429502 IC50 = 1.6 nM T40016 C37VXR 10432143 Ki = 3210 nM T40016 CAKV91 10434383 IC50 = 10 nM T40016 CFMI34 10440737 IC50 = 310 nM T40016 C1KE6C 10446402 IC50 = 2600 nM T40016 CI91JZ 10450619 IC50 = 1000 nM T40016 CK05HV 10450738 IC50 = 167 nM T40016 CT35HI 10452933 EC50 = 38 nM T40016 CS12VO 10453115 EC50 = 6 nM T40016 C0NT9D 10454007 IC50 = 5.3 nM T40016 CVQS04 10454813 IC50 = 6.7 nM T40016 CH49LB 10456872 EC50 = 24.2 nM T40016 C9LQ7R 10457600 IC50 = 5.012 nM T40016 C7R2OJ 10457897 IC50 = 5.012 nM T40016 C1H5RP 10458842 EC50 > 10 nM T40016 CYQ65Z 10472575 IC50 = 125 nM T40016 CK4NI1 10473865 IC50 = 280 nM T40016 COMX74 10474093 IC50 = 1.2 nM T40016 C85RBN 10474264 IC50 = 190 nM T40016 C1S9HE 10474749 IC50 = 395 nM T40016 CUL8O4 10475384 EC50 = 2.9 nM T40016 CN7KQ8 10475688 IC50 = 371 nM T40016 CGH31Z 10475742 EC50 = 1 nM T40016 C8O1QG 10476314 Ki = 913 nM T40016 CPX65M 10477088 IC50 = 64 nM T40016 CG3P0I 10478173 EC50 = 31.3 nM T40016 C5U3JY 10478638 IC50 = 5.1 nM T40016 CB3S1Q 10484201 IC50 = 2.1 nM T40016 CYE7C2 10496255 Ki = 3697 nM T40016 CT7IG5 10497270 Ki = 1657 nM T40016 CO35TR 10499308 Ki = 6386 nM T40016 C6FA1N 10501542 Ki = 2570 nM T40016 CA5OH2 10503046 Ki = 14 nM T40016 C5AP6C 10503520 Ki = 42 nM T40016 C5WP1Q 10517398 Ki = 8511 nM T40016 CR1OS9 10523126 Ki = 909 nM T40016 C5CDF0 10524606 Ki = 4109 nM T40016 CYS8J9 10546095 Ki > 10000 nM T40016 CB04AE 10593144 Ki = 2206 nM T40016 CBEC38 10596252 Ki = 60 nM T40016 C6G7JR 10596379 Ki = 193 nM T40016 CC8T7J 10598305 Ki = 59 nM T40016 CAD6L2 10618033 Ki = 1036 nM T40016 CMK8I6 10622122 Ki = 6.3 nM T40016 CO3V0S 10622594 Ki = 67 nM T40016 C57PFY 10643931 Ki = 864 nM T40016 C02ZMG 10643956 Ki = 58 nM T40016 CF08PC 10661117 Ki = 8215 nM T40016 CU9X3A 10665612 Ki = 1261 nM T40016 C69CNF 10667548 Ki = 680 nM T40016 CYNG45 10668755 Ki = 173 nM T40016 CS6YF0 10690456 Ki = 249 nM T40016 CYRQ10 10691647 Ki = 9.3 nM T40016 C6SP3O 10694256 Ki = 257 nM T40016 CVD2Y9 10717098 Ki = 100 nM T40016 CK2NM9 10717832 Ki = 250 nM T40016 CUG2Z9 10739308 Ki = 2199 nM T40016 CAT1X8 10741366 Ki = 34 nM T40016 C3H6CZ 10754393 Ki = 8356 nM T40016 CB3JD0 10763832 Ki = 39 nM T40016 C7HAB1 10782276 Ki = 4532 nM T40016 CNV27D 10783127 Ki = 2781 nM T40016 CNL1U7 10785305 Ki > 10000 nM T40016 C07BOR 10787258 Ki = 147 nM T40016 C10AMX 10805958 Ki = 2286 nM T40016 CBX48C 10807828 Ki = 2670 nM T40016 CN5WV4 10809583 Ki = 4417 nM T40016 C1CRQ5 10811045 Ki = 237 nM T40016 CL7JN6 10827013 Ki = 6812 nM T40016 CN1H5Z 10832792 Ki = 80 nM T40016 CA96PR 10860931 Ki = 7 nM T40016 C8KME1 10861665 Ki = 88 nM T40016 CHU9A4 10873317 IC50 = 77 nM T40016 CI5F0S 10881662 Ki = 33.8 nM T40016 CVG34R 10883247 Ki = 34 nM T40016 CK41RM 10892050 Ki > 10000 nM T40016 CNG7L9 10894018 Ki = 4.2 nM T40016 CP9FX4 10904951 Ki = 3200 nM T40016 C54IAT 10905085 Ki = 1800 nM T40016 C6EG2D 10906030 Ki = 5.32 nM T40016 CBD12K 10906044 IC50 = 320 nM T40016 C3BZD9 10916860 Ki = 6000 nM T40016 C1D8IK 10926892 Ki = 400 nM T40016 C2UG0A 10937849 Ki = 207 nM T40016 C2IJR9 10949091 Ki = 2100 nM T40016 CHU10G 10960295 Ki = 232 nM T40016 CT2BR8 10969959 Ki = 4.4 nM T40016 C0GX6P 10970905 Ki = 25 nM T40016 CV3QY8 10972344 Ki = 2.3 nM T40016 C07JFA 10993685 Ki = 386 nM T40016 CUC05J 11002535 Ki = 2.3 nM T40016 C8AY9Z 11003946 Ki = 51 nM T40016 C5U8ZE 11013870 Ki = 18 nM T40016 CMJ7F9 11013871 Ki = 2 nM T40016 C7E9XI 11015162 IC50 = 90 nM T40016 CRH3L8 11025398 IC50 = 250 nM T40016 CU02DM 11046701 Ki = 5.2 nM T40016 CF8UC7 11057125 Ki = 140 nM T40016 CUYB81 11057924 Ki = 6.6 nM T40016 CIH8K4 11066740 Ki = 5.96 nM T40016 CS7Q4F 11069511 Ki = 2.8 nM T40016 CI8GJ5 11079263 IC50 = 109 nM T40016 C09ZLY 11088436 Ki > 10000 nM T40016 C6T7CR 11089159 Ki = 9.3 nM T40016 C6HPL0 11089468 Ki = 1.9 nM T40016 C6LYG7 11090322 IC50 > 1000 nM T40016 CE2O8Y 11110616 Ki = 6.9 nM T40016 C69GXQ 11110815 Ki = 9 nM T40016 CDX2W3 11121575 Ki = 18 nM T40016 C1OJK3 11131414 Ki = 27.6 nM T40016 CBDG76 11132271 Ki > 5000 nM T40016 C6TJ8D 11132273 Ki = 3.8 nM T40016 CB03TK 11143041 EC50 = 99700 nM T40016 CXS6J7 11155441 Ki = 0.2 nM T40016 CJ7KZ9 11155655 Ki > 100000 nM T40016 CIX9T7 11177172 EC50 = 54.2 nM T40016 CP3D7X 11201812 IC50 = 10 nM T40016 CW0Z2J 11212626 IC50 = 4786.3 nM T40016 CL97OU 11212803 IC50 = 17 nM T40016 C4U0DF 11213029 EC50 = 0.2 nM T40016 CFH3Q8 11213179 Ki = 2.9 nM T40016 C81CJV 11214068 IC50 = 0.5 nM T40016 CLCM91 11224044 IC50 = 0.9 nM T40016 CF3AY1 11225369 IC50 = 3 nM T40016 CVR9L1 11226313 EC50 = 0.5 nM T40016 CRN4V2 11232136 IC50 > 3000 nM T40016 CW6P7A 11244720 EC50 = 3 nM T40016 C3DO9S 11248612 IC50 = 2.5 nM T40016 CYCR06 11256303 IC50 = 14 nM T40016 CXG0C2 11269006 IC50 = 1.5 nM T40016 C8XPZ4 11269445 IC50 = 57 nM T40016 C4HNB8 11269886 IC50 = 22 nM T40016 CSH2R3 11271731 EC50 = 4.5 nM T40016 CHXY45 11272042 EC50 = 0.4 nM T40016 CJLC62 11273833 IC50 = 330 nM T40016 CC0XI4 11279959 IC50 = 127 nM T40016 C4SC0W 11281576 EC50 = 2.2 nM T40016 C8YL6K 11282486 IC50 = 19 nM T40016 CUX0S2 11282904 Ki = 0.6 nM T40016 CIY9H5 11291999 IC50 = 6 nM T40016 C58MZD 11293264 IC50 = 0.4 nM T40016 C8UK5D 11302609 IC50 = 38 nM T40016 C24ILB 11302908 Ki = 2250 nM T40016 C0IQ9K 11304445 IC50 = 4 nM T40016 CLIB17 11304952 EC50 = 0.6 nM T40016 C0XUF2 11305564 IC50 = 1.9 nM T40016 C5C0MA 11316115 IC50 = 2.5 nM T40016 C0B2FT 11327284 IC50 = 5 nM T40016 CXC9G3 11327341 IC50 = 1400 nM T40016 C3OI8M 11330644 IC50 = 6.6 nM T40016 C1HZS7 11336351 IC50 = 73 nM T40016 CT9Y4O 11339440 IC50 > 3000 nM T40016 CGM2R9 11339795 IC50 = 562.34 nM T40016 CBPX74 11350176 IC50 = 26 nM T40016 CQ1NV4 11363810 Ki = 1.5 nM T40016 CUE7W0 11375176 EC50 = 1.5 nM T40016 C8FQ9B 11375180 IC50 = 2090 nM T40016 CP2DL0 11377050 IC50 = 500 nM T40016 C76VYN 11382721 IC50 = 230 nM T40016 CV4RO2 11384310 IC50 = 2 nM T40016 CXW40M 11384346 IC50 = 9 nM T40016 CU7IE0 11410199 IC50 = 5.4 nM T40016 CO20QH 11416730 IC50 = 120 nM T40016 C5KQY8 11417666 Ki = 225 nM T40016 C5WO0U 11429662 EC50 = 6.5 nM T40016 C8DXS2 11430241 EC50 = 0.7 nM T40016 CSGJ21 11430586 Ki = 1.9 nM T40016 C2D7HP 11442368 IC50 = 22 nM T40016 COQ7S4 11444087 Ki = 0.9 nM T40016 CV8XI7 11453933 EC50 = 0.6 nM T40016 C2BXU1 11454745 Ki = 4.3 nM T40016 C8Y5BF 11463839 EC50 = 19.5 nM T40016 CJEU23 11474124 IC50 = 77.3 nM T40016 CD2Q3F 11474917 IC50 = 3 nM T40016 CAT79U 11475733 EC50 = 1.9 nM T40016 CC75NQ 11477616 Ki = 0.6 nM T40016 CQ62KS 11485693 IC50 = 190 nM T40016 C9Q1NY 11494167 Ki = 1.3 nM T40016 CFLQ08 11495227 IC50 = 8.2 nM T40016 C03NYX 11495549 IC50 = 210 nM T40016 CJ1M8L 11495854 Ki = 17 nM T40016 CFB75K 11497883 Ki = 4.5 nM T40016 CK3RS0 11498018 Ki = 12 nM T40016 C0O7TM 11500993 Ki = 100 nM T40016 C3L4DF 11504875 EC50 = 75000 nM T40016 CR40IH 11516847 IC50 = 8 nM T40016 C4Q5XE 11517391 Ki = 6 nM T40016 CP4F8X 11517412 IC50 = 2.3 nM T40016 CB9D3A 11517558 IC50 = 11.22 nM T40016 CCL20N 11519406 Ki = 3 nM T40016 CS0M3B 11525591 Ki = 1.1 nM T40016 CE3I6O 11525793 IC50 = 12.59 nM T40016 C2PB6Z 11530605 Ki = 8 nM T40016 C1R6DC 11531942 IC50 = 37 nM T40016 C9SH1C 11532777 IC50 = 31.62 nM T40016 C0DS3E 11533163 Ki = 2.6 nM T40016 C7F0KV 11533276 IC50 = 19.95 nM T40016 CZ1HA3 11538472 IC50 = 16 nM T40016 CFC1Z4 11538799 IC50 = 26 nM T40016 C16YOG 11541310 Ki = 1.4 nM T40016 CNRP26 11545475 IC50 = 18 nM T40016 C8YBI3 11547009 Ki = 13 nM T40016 CP13VG 11547261 Ki = 41 nM T40016 CT45RM 11548068 IC50 = 1.202 nM T40016 CI90JB 11551816 IC50 = 10 nM T40016 C0J8UL 11551817 Ki = 4.4 nM T40016 C4FM3R 11553707 IC50 = 1.259 nM T40016 CBK60G 11559947 IC50 = 23 nM T40016 C1D9YS 11560003 IC50 = 15 nM T40016 C1XKY3 11561826 Ki = 18 nM T40016 C47ROU 11562491 Ki = 0.8 nM T40016 CB37YF 11566981 Ki = 1.8 nM T40016 C5UEY6 11567352 IC50 = 2.1 nM T40016 C8WJ2F 11567609 IC50 = 4.5 nM T40016 CXQ59S 11567630 IC50 = 99 nM T40016 C0PES1 11568433 IC50 = 1.95 nM T40016 CJ30TW 11568951 Ki = 2.5 nM T40016 C0QFC2 11569557 Ki = 12 nM T40016 CQ28XT 11569834 Ki = 0.6 nM T40016 C10AWO 11569892 IC50 = 794.33 nM T40016 C7AMJ5 11570728 Ki = 1.3 nM T40016 C1X7LS 11571692 EC50 = 50 nM T40016 CQ0U9D 11576238 IC50 = 25.12 nM T40016 CSQ32L 11577390 Ki = 1.4 nM T40016 CTA8J3 11583514 IC50 = 15.85 nM T40016 CQ43OD 11584668 Ki = 2.8 nM T40016 CEF7K8 11585049 EC50 = 173000 nM T40016 C0SCT6 11588584 IC50 = 31 nM T40016 C3MW1D 11589982 IC50 = 7.1 nM T40016 C03QYZ 11590471 IC50 = 15 nM T40016 CLN0C5 11591199 IC50 = 9.55 nM T40016 CZ4M8O 11591459 IC50 = 3.467 nM T40016 CEH7D2 11591552 Ki = 0.6 nM T40016 CV94WU 11591790 Ki = 26 nM T40016 CZO0L1 11595527 Ki = 5.8 nM T40016 CAO2P1 11596392 IC50 = 17 nM T40016 CJWP94 11596794 EC50 = 8.318 nM T40016 C53OBJ 11597965 Ki = 22 nM T40016 C54HCR 11598367 IC50 = 12.59 nM T40016 C3FJQ8 11602375 IC50 = 35000 nM T40016 C8RO4G 11611666 IC50 = 0.5012 nM T40016 C7PS2W 11612527 IC50 = 15.85 nM T40016 C7ME6V 11613022 IC50 = 9.55 nM T40016 CC0I2P 11613420 IC50 = 8.511 nM T40016 CSB97O 11617028 Ki = 0.3 nM T40016 CC49FR 11617298 Ki = 79 nM T40016 CR5DA0 11617684 Ki = 24 nM T40016 CI1D2W 11620916 Ki = 0.8 nM T40016 C1IEC7 11627493 IC50 = 11.48 nM T40016 CRF4E1 11631740 EC50 = 0.8 nM T40016 CW6R3T 11631784 Ki = 0.8 nM T40016 CRL3A7 11632925 IC50 = 25 nM T40016 CQB0E3 11633482 IC50 = 15 nM T40016 C9DNG1 11640164 IC50 = 4 nM T40016 CC4LE3 11640246 IC50 = 3.09 nM T40016 CB4E0S 11645780 Ki = 460 nM T40016 C3MHY7 11646048 IC50 = 5.3 nM T40016 C1RJ3I 11646689 IC50 = 9 nM T40016 CX3L5S 11647533 IC50 = 18 nM T40016 C2AD9C 11647851 Ki = 10 nM T40016 CU3K9V 11653520 Ki = 4.5 nM T40016 C4S5RG 11655053 IC50 = 34 nM T40016 C5L3GN 11656415 Ki = 1.6 nM T40016 CDOZ32 11661172 IC50 = 10 nM T40016 C1CEJ0 11663141 EC50 = 18.62 nM T40016 CEQR07 11663523 EC50 = 17.78 nM T40016 CH8F5J 11663592 IC50 = 5.012 nM T40016 C0LEZ3 11667800 IC50 = 14 nM T40016 C5XEN0 11668719 IC50 = 340 nM T40016 CCWJ64 11668984 IC50 = 48 nM T40016 CTE80K 11671653 Ki = 8.6 nM T40016 CM57PA 11682250 IC50 = 12 nM T40016 CZPK72 11682989 IC50 = 15 nM T40016 C1HA4U 11684596 IC50 = 125.89 nM T40016 C4QA6V 11685011 IC50 = 6.31 nM T40016 C8SY4D 11688929 Ki = 90 nM T40016 CCK83U 11690269 IC50 = 8 nM T40016 CH7I6J 11691206 IC50 = 12.59 nM T40016 CY07JH 11696378 IC50 = 51 nM T40016 CBU02W 11696959 IC50 = 4 nM T40016 C2S9IT 11697271 IC50 = 13 nM T40016 CGR32I 11697882 IC50 = 5 nM T40016 C42NIT 11697950 Ki = 340 nM T40016 C25NSM 11699191 IC50 = 8.128 nM T40016 C7VC2U 11699294 IC50 = 1380.38 nM T40016 C3OQH4 11703401 IC50 = 67 nM T40016 C75IBX 11704529 IC50 = 20 nM T40016 CGX54N 11704756 IC50 = 320 nM T40016 CI4JW3 11706478 Ki = 0.9 nM T40016 CO2N1W 11710364 IC50 = 9 nM T40016 C8OPA1 11710962 IC50 = 19 nM T40016 CW3N8H 11711766 IC50 = 280 nM T40016 C1TQX9 11712150 Ki = 15 nM T40016 C6AB0O 11712629 IC50 = 16.6 nM T40016 COEU05 11719039 IC50 = 60 nM T40016 CM3BG2 11724520 IC50 > 2000 nM T40016 C4OH1Y 11726899 Ki > 10000 nM T40016 C0VJ3I 11727825 Ki > 5000 nM T40016 CVA1S3 11728656 Ki = 5.42 nM T40016 CZ0B7H 11731863 Ki = 84 nM T40016 CYJ73N 11733546 IC50 = 40.9 nM T40016 CQO76Z 11741168 IC50 = 1400 nM T40016 CJC5A2 11741840 IC50 = 4.2 nM T40016 C87YNC 11741891 IC50 = 22 nM T40016 CH92VI 11743259 IC50 = 15 nM T40016 CV49MT 11747706 IC50 = 133 nM T40016 C5HLU8 11750204 IC50 = 1.4 nM T40016 C9UED8 11752131 EC50 = 0.2 nM T40016 CY1F4I 11752649 EC50 = 0.2 nM T40016 C3XF4G 11755231 IC50 = 7.943 nM T40016 CKD9R8 11757239 IC50 = 9.2 nM T40016 CEWP04 11771756 IC50 = 8.8 nM T40016 CQU0E7 11774868 IC50 = 14 nM T40016 COI0P1 11774981 IC50 = 510 nM T40016 CR70FP 11794088 Ki = 2379 nM T40016 CU7EJ1 11822858 Ki = 157 nM T40016 C5FRJ6 11825145 Ki = 18 nM T40016 C4U8KY 12085089 IC50 = 2 nM T40016 CEV10S 13278723 IC50 = 1.8 nM T40016 C7ICM3 15298636 IC50 = 18 nM T40016 C14LTD 15463551 IC50 = 10 nM T40016 CC15FW 16049465 IC50 = 2.3 nM T40016 CMZH47 16051364 IC50 > 10000 nM T40016 C3QOV0 16099227 IC50 = 10 nM T40016 CW6LO1 16099229 IC50 > 2000 nM T40016 C2R4PK 16099231 IC50 = 38 nM T40016 C9KM7X 16099232 IC50 = 120 nM T40016 C05CYN 16099234 IC50 = 950 nM T40016 CJQ8A1 16099236 IC50 = 6 nM T40016 CA72YW 16099237 IC50 = 780 nM T40016 CS07DB 16099238 IC50 = 4 nM T40016 C42ESN 16099240 IC50 = 5 nM T40016 CMZ91J 16099242 IC50 > 2000 nM T40016 CF69RC 16099243 IC50 > 2000 nM T40016 C60GEM 16099245 IC50 = 110 nM T40016 CE48CS 16099246 IC50 = 650 nM T40016 CTF2M7 16099247 IC50 = 4 nM T40016 CX9BK2 16099248 IC50 = 54 nM T40016 CN6PA9 16099249 IC50 = 28 nM T40016 C9Z6AK 16099250 IC50 = 10 nM T40016 C5Z8HR 16099251 IC50 = 11 nM T40016 CWK76M 16099252 IC50 = 3 nM T40016 CU1YV4 16099253 IC50 = 34 nM T40016 CN5VS8 16099254 IC50 = 125 nM T40016 CC24LB 16110489 EC50 > 10 nM T40016 C3BU9M 16216822 IC50 = 29 nM T40016 C1Q5SV 16220168 IC50 = 5600 nM T40016 CH6CN0 16658901 Ki = 8500 nM T40016 CU9LS2 16661702 EC50 = 7900 nM T40016 C9F2VT 16665286 IC50 = 3.9 nM T40016 C2H9EM 16665289 IC50 = 6.9 nM T40016 CT6Y5F 16665374 IC50 = 3.4 nM T40016 CI95KE 16665449 IC50 = 9.7 nM T40016 CYW0T9 16665451 IC50 = 12 nM T40016 CP8VM0 16665452 IC50 = 23 nM T40016 CPNJ02 16665453 IC50 = 5.7 nM T40016 C0OG7T 16665528 IC50 = 16 nM T40016 CMC9W0 16665533 IC50 = 12 nM T40016 CV3OM1 16665605 IC50 = 7.7 nM T40016 CCN5F6 16665606 IC50 = 795 nM T40016 CG5UM0 16665608 IC50 = 12 nM T40016 CLJ2U5 16666385 IC50 = 5.2 nM T40016 C1UY8J 16666386 IC50 = 1.47 nM T40016 CWR10T 16666470 IC50 = 5.4 nM T40016 CWEJ30 16666472 IC50 = 1.5 nM T40016 C0Y2OK 16721017 IC50 = 304 nM T40016 CE71BC 16722203 IC50 = 37.6 nM T40016 C92NRU 16727109 EC50 > 25000 nM T40016 CF6V2J 16730097 IC50 = 111 nM T40016 CWK35C 16730429 IC50 = 14000 nM T40016 C9BC0L 16732000 Ki > 10000 nM T40016 CLC2Z8 16739323 IC50 = 86.5 nM T40016 CAL7M5 16756781 IC50 = 34000 nM T40016 C3RPY2 17747503 IC50 = 6.3 nM T40016 CLNU15 17758014 EC50 = 0.2 nM T40016 C62WRI 17758132 EC50 = 0.2 nM T40016 C5GRB8 17758133 EC50 = 0.4 nM T40016 CSKX58 17758233 Ki = 1.2 nM T40016 C7CPW9 17758234 EC50 = 0.1 nM T40016 CI5KT6 17758236 EC50 = 0.5 nM T40016 CE8C5G 17758459 IC50 = 1 nM T40016 C32WCP 17758569 EC50 = 0.6 nM T40016 C05ARI 17758570 EC50 = 1.4 nM T40016 CX03YG 18188955 IC50 = 2 nM T40016 CQLU68 18189214 IC50 = 402 nM T40016 CH39OX 18504012 IC50 = 48 nM T40016 CYZ71G 18511908 IC50 = 370 nM T40016 C7ZIF9 18511910 IC50 = 2.9 nM T40016 CEFA90 18511931 IC50 = 34 nM T40016 CEDU50 18511945 IC50 = 96 nM T40016 C4EU2J 18511975 IC50 = 470 nM T40016 CL91CU 18511977 IC50 = 14 nM T40016 CQ4BF7 18511980 IC50 = 100 nM T40016 C9C8GH 18511994 IC50 = 48 nM T40016 CZO79P 18512002 IC50 = 58 nM T40016 C05YOA 18512008 IC50 = 56 nM T40016 C03SPA 18512022 IC50 = 47 nM T40016 CR5G8F 18512030 IC50 = 63 nM T40016 C7LFU4 18512032 IC50 = 320 nM T40016 CF6E2C 18512049 IC50 = 26 nM T40016 C1ZVD4 18512058 IC50 = 17 nM T40016 CGJ56E 18512087 IC50 = 36 nM T40016 C0C6BG 18512103 IC50 = 11 nM T40016 C49PLT 18512117 IC50 = 138 nM T40016 CX3B4O 18512130 IC50 = 3.9 nM T40016 C3C7ID 18512158 IC50 = 5.4 nM T40016 CJCF08 18512161 IC50 = 270 nM T40016 C7XC4K 18512162 IC50 = 1.4 nM T40016 C5YX7A 18512163 IC50 = 250 nM T40016 CR19ST 18512166 IC50 = 28 nM T40016 CB5C3I 18512168 IC50 = 11 nM T40016 CFI8E1 18512170 IC50 = 15 nM T40016 CM4B9R 18512171 IC50 = 220 nM T40016 CRP45C 18512178 IC50 = 1000 nM T40016 C64PAE 18512192 IC50 = 13 nM T40016 C14RFT 18512213 IC50 = 8.8 nM T40016 CTX2Z5 18512224 IC50 = 21 nM T40016 CL42KX 18512282 IC50 = 290 nM T40016 CX1FQ2 18512329 IC50 = 2.4 nM T40016 CEN14G 18512334 IC50 = 5.7 nM T40016 CD8JC6 18512366 IC50 = 120 nM T40016 CJG26V 18512380 IC50 = 1.5 nM T40016 CLX02Q 18512392 IC50 = 2.7 nM T40016 CXM9D1 18512399 IC50 = 60 nM T40016 CS9CI5 18551230 EC50 = 45 nM T40016 CBI64N 18551237 IC50 = 8 nM T40016 CLUA26 18551266 IC50 = 230 nM T40016 C5ZYJ0 20231824 Ki = 50 nM T40016 CEH7V5 20786216 IC50 = 6.31 nM T40016 CR73OM 21136439 IC50 = 892 nM T40016 CF0S6J 21210483 IC50 = 11700 nM T40016 C97WCO 21941658 EC50 = 10 nM T40016 CCI89R 21948853 IC50 = 1.995 nM T40016 CB2SF4 21948904 IC50 = 3.162 nM T40016 CP7S2I 21970730 IC50 = 289 nM T40016 C2ZP7V 22218142 IC50 > 10000 nM T40016 CWA9Q6 22284899 IC50 = 760 nM T40016 CY5Z4Q 22314851 IC50 = 13 nM T40016 C5N1HK 22314910 IC50 > 5000 nM T40016 C6R1WN 22314926 IC50 = 42 nM T40016 CDQ10L 22314947 IC50 = 150 nM T40016 C8XAR4 22314951 IC50 = 220 nM T40016 C84QJV 22314968 IC50 = 12 nM T40016 C4I7OB 22314982 IC50 = 23 nM T40016 CGWM75 22315021 IC50 = 320 nM T40016 C1GIZ6 22315043 IC50 = 20 nM T40016 C1QTK4 22398492 IC50 = 7 nM T40016 C6CSB4 22398502 IC50 = 160 nM T40016 CR8N1E 22398506 IC50 = 27 nM T40016 CM83TU 22398533 IC50 = 8 nM T40016 C34LHW 22398559 IC50 = 21 nM T40016 CJBW90 22398592 IC50 = 23 nM T40016 CEJ65O 22398627 IC50 = 8 nM T40016 CCYS56 22566499 IC50 = 303 nM T40016 CGE03P 22566506 IC50 = 260 nM T40016 CH29BV 22566507 IC50 = 116 nM T40016 C21YKI 22566509 IC50 = 404 nM T40016 CU8D7L 22566515 IC50 > 2000 nM T40016 CPQ9O5 22605977 IC50 = 2100 nM T40016 CCF52I 22605979 IC50 > 2000 nM T40016 CGY94Z 23433542 IC50 = 3200 nM T40016 CZ9L3J 23552303 IC50 = 87 nM T40016 CL0H7I 23595919 Ki = 303 nM T40016 C56STL 23595942 EC50 = 330.6 nM T40016 CP9SN1 23596227 Ki = 92.6 nM T40016 CNVC31 23596254 Ki = 82.5 nM T40016 C9O6RB 23596322 Ki = 4.1 nM T40016 CNLR52 23596329 Ki = 8.7 nM T40016 CMV6U7 23596330 Ki = 22.6 nM T40016 C4F7OG 23596337 Ki = 3.9 nM T40016 CJ0XR3 23625602 IC50 = 1.585 nM T40016 CF4UA3 23648072 IC50 = 1060 nM T40016 CSV4D3 23648197 EC50 = 19 nM T40016 CBI6J3 23648200 EC50 = 3 nM T40016 CT80JO 23648203 EC50 = 46 nM T40016 CD74QP 23648204 EC50 = 32 nM T40016 CHW3X2 23648205 EC50 = 3 nM T40016 C0VE5H 23648206 EC50 = 5 nM T40016 C7BLN0 23992759 Ki = 157.7 nM T40016 CWPH96 24180508 IC50 = 99 nM T40016 CS1KX2 24180659 Ki = 14 nM T40016 CZI4C6 24739672 Ki = 1860 nM T40016 CS23KY 24739834 Ki = 977 nM T40016 C1M9QG 24739836 Ki = 927 nM T40016 CG5SJ0 24739997 Ki = 1530 nM T40016 C7Z1HW 24740156 Ki = 780 nM T40016 CTE1N2 24748569 EC50 > 10000 nM T40016 CQ57SD 24748957 IC50 = 48.98 nM T40016 CWL9G2 24748958 IC50 = 8.128 nM T40016 C14ZOJ 24748959 EC50 = 41.69 nM T40016 CSP7E5 24748960 EC50 = 61.66 nM T40016 C8J3HZ 24748961 IC50 = 6.607 nM T40016 CXAJ63 24749047 IC50 = 7.244 nM T40016 CAS4V3 24749048 IC50 = 8.913 nM T40016 C6TAE7 24749049 IC50 = 1.585 nM T40016 C36ECZ 24749050 IC50 = 30.2 nM T40016 CMBK68 24749150 IC50 = 147.91 nM T40016 C7ZU9P 24749151 EC50 = 12.88 nM T40016 C4WYE7 24749678 Ki = 167 nM T40016 CY2JS4 24749684 Ki = 54.4 nM T40016 C2QHO3 24749808 Ki = 5.93 nM T40016 CR1G7M 24768971 EC50 = 3.981 nM T40016 CM8Y4V 24769095 IC50 = 0.7943 nM T40016 C5S6JN 24780149 IC50 = 6.31 nM T40016 CW5TJ7 24781731 IC50 = 15.85 nM T40016 CPVS80 24789142 EC50 = 4.1 nM T40016 C8OCU9 24789150 Ki = 1 nM T40016 CR48VC 24809711 EC50 = 7.943 nM T40016 CGC0D7 24816319 IC50 = 11 nM T40016 CNM45B 24850992 IC50 = 1510 nM T40016 C1JTW2 24851053 Ki = 0.257 nM T40016 CC53XL 24860583 Ki = 15 nM T40016 C5Y2TN 24873449 IC50 = 0.69 nM T40016 CGE0V4 24882669 IC50 = 10 nM T40016 C58RHY 24883011 IC50 = 2500 nM T40016 CW35CK 24883012 IC50 = 1800 nM T40016 C3SC0V 24883054 IC50 = 1700 nM T40016 C4SA6C 24883055 IC50 = 470 nM T40016 C5LZK2 24895096 IC50 = 34 nM T40016 CMH52V 24936311 Ki = 0.53 nM T40016 CA3O5Q 24936312 Ki = 10.2 nM T40016 COGP96 24936313 Ki = 5.14 nM T40016 C5WOB6 24936314 Ki = 0.72 nM T40016 CM8NR9 24936446 Ki = 1.74 nM T40016 CVY09S 24936449 Ki = 0.64 nM T40016 CD8JT0 24936598 Ki = 11 nM T40016 CT8L2W 24936727 Ki = 14 nM T40016 CFK6W8 24936729 Ki = 11 nM T40016 C1BR3F 24936732 Ki = 18 nM T40016 CBN24H 24936982 Ki = 1.7 nM T40016 C71KJS 24936984 Ki = 2.4 nM T40016 C65YPH 24937240 Ki = 5.7 nM T40016 C7YCB3 24937242 Ki = 12 nM T40016 C26TWN 24937362 Ki = 5 nM T40016 C26HUZ 24937363 EC50 = 10 nM T40016 CEV09L 24937493 Ki = 2.4 nM T40016 CZ91CN 24937934 IC50 = 0.3162 nM T40016 C4YTH3 24937935 IC50 = 0.1259 nM T40016 C9KFD4 24937936 IC50 = 0.07943 nM T40016 CXTL09 24945221 Ki = 2 nM T40016 CQFZ96 24945227 Ki = 3 nM T40016 CQ2FL3 24945386 Ki = 2 nM T40016 C5DW7P 24945389 Ki = 1 nM T40016 CTV40U 24945468 Ki = 4 nM T40016 CV03UT 24945548 Ki < 1 nM T40016 CYL54C 24945619 Ki < 1 nM T40016 C8L9PC 24945705 Ki = 10 nM T40016 C06PDG 24952192 Ki = 0.3 nM T40016 CG1CF9 24952193 Ki = 0.8 nM T40016 CZC7L8 24953162 IC50 = 0.91 nM T40016 C1CUZ4 24953163 IC50 = 13 nM T40016 CZB7M8 24953166 IC50 = 7.4 nM T40016 CU3A7E 24953513 IC50 = 37 nM T40016 CKML07 24954062 Ki = 1 nM T40016 C07FUV 24954066 Ki = 13 nM T40016 CP1G9U 24954421 Ki = 4 nM T40016 CNJS10 24954422 Ki = 169 nM T40016 CC4P9R 24954791 Ki = 2 nM T40016 CSD27Y 24954792 Ki = 4 nM T40016 CW7O3D 24954793 Ki = 4 nM T40016 CZ14BO 24954794 Ki = 2 nM T40016 C4W7BN 24954947 IC50 = 0.75 nM T40016 C6XC2R 24954951 IC50 = 1.4 nM T40016 CFK32R 24955041 Ki = 6 nM T40016 CL70XN 24955148 Ki = 2 nM T40016 CN9L1B 24955149 Ki = 1 nM T40016 CLJ87T 24955150 Ki = 8 nM T40016 CK96WS 24955151 Ki = 5 nM T40016 CVU18K 24955152 Ki = 5 nM T40016 CRBW74 24956466 Ki = 412 nM T40016 CYES17 24957737 Ki = 55 nM T40016 C85BHZ 24958028 IC50 = 12.59 nM T40016 C3VO7Q 24960588 EC50 = 39.81 nM T40016 C83YKB 24961057 Ki = 11 nM T40016 CQ3X6G 24961686 EC50 = 25.12 nM T40016 CZ89IP 24961687 EC50 = 6.31 nM T40016 CZG93W 24961689 EC50 = 251.19 nM T40016 CLY07O 24961690 EC50 = 50.12 nM T40016 C42YHP 24962051 IC50 = 316.23 nM T40016 C5W1IT 24962055 IC50 = 19.95 nM T40016 CN49EG 24962146 Ki = 151 nM T40016 CYEF46 24964075 Ki < 1 nM T40016 CVI3O1 24964440 Ki = 2 nM T40016 CS7WY4 24964443 Ki < 1 nM T40016 CIGM27 24983460 IC50 = 20 nM T40016 CP1VY8 24997743 IC50 = 98 nM T40016 CM2Z0U 25011854 IC50 = 0.66 nM T40016 CX7I2K 25012028 IC50 = 4.6 nM T40016 CR7GA9 25012190 IC50 = 0.05 nM T40016 CO9S6B 25013321 IC50 = 0.62 nM T40016 CHY0D7 25013322 IC50 = 0.13 nM T40016 C0J3CQ 25013326 IC50 = 0.25 nM T40016 CZE7X8 25013489 IC50 = 0.21 nM T40016 CAF85M 25013490 IC50 = 0.08 nM T40016 C0TPS5 25013653 IC50 = 2.9 nM T40016 CHN41A 25013654 IC50 = 0.03 nM T40016 CWU91M 25013811 EC50 = 1.3 nM T40016 CSH29L 25013812 IC50 = 0.04 nM T40016 C68SGK 25014203 IC50 = 3.1 nM T40016 C6SA2C 25014204 IC50 = 5.09 nM T40016 CKUA52 25014206 IC50 = 1.41 nM T40016 C0LO9C 25028373 EC50 = 50.12 nM T40016 C4H7UP 25048180 IC50 = 4100 nM T40016 C2G1JK 25053351 Ki > 30000 nM T40016 CAW8M0 25070694 IC50 > 3000 nM T40016 C3H0KR 25110774 Ki = 0.6 nM T40016 C4GLY1 25110785 Ki = 1.4 nM T40016 CCL91F 25110786 Ki = 0.8 nM T40016 C21XDY 25145083 Ki > 10000 nM T40016 CS6JQ1 25167502 Ki = 1.5 nM T40016 C0XPW9 25168896 IC50 = 210 nM T40016 CUL27D 25168900 IC50 = 95 nM T40016 CEV2D7 25205475 IC50 = 2 nM T40016 C9S0ZW 25205477 IC50 = 7 nM T40016 C49KHR 25206116 IC50 = 2 nM T40016 C87ZHT 25231296 IC50 = 0.9 nM T40016 CLY9W3 25235364 IC50 = 1.5 nM T40016 C3FW0Y 25257459 IC50 = 360 nM T40016 CVO06A 25257700 IC50 = 1100 nM T40016 CN03HI 25257925 IC50 = 17 nM T40016 CY6X2V 25258136 IC50 = 5.6 nM T40016 CS49WQ 25258137 IC50 = 3.5 nM T40016 CV4Y6N 25258138 IC50 = 6.2 nM T40016 C5NGC7 25258139 IC50 = 1.5 nM T40016 C1OJ6Z 25258140 IC50 > 1000 nM T40016 CWT31Y 25258141 IC50 > 1000 nM T40016 CJ68WY 25258142 IC50 = 21 nM T40016 CLX0P9 25258381 IC50 = 2.3 nM T40016 CM48WL 25258382 IC50 = 1500 nM T40016 CNLS64 25258386 IC50 = 2.5 nM T40016 CSG7P9 25258611 IC50 = 3 nM T40016 CN87ME 25258614 IC50 = 3.8 nM T40016 CX89HM 44138106 Ki = 1 nM T40016 C9LCJ5 44156980 IC50 = 4.8 nM T40016 CZAJ06 44193143 Ki = 6.2 nM T40016 CS36WU 44193144 Ki = 7.6 nM T40016 CXZ35T 44193145 Ki = 6.8 nM T40016 C2MOF7 44193146 Ki = 7.8 nM T40016 CWR6X1 44193147 Ki = 4.3 nM T40016 CF02JG 44193242 Ki = 14.3 nM T40016 C3JOW4 44193245 IC50 = 13 nM T40016 C9WB1Z 44193246 Ki = 16.1 nM T40016 CKDG10 44193342 Ki = 70 nM T40016 C4Q0SG 44193344 IC50 = 7.5 nM T40016 CK9ZL7 44193440 EC50 = 3.5 nM T40016 CYE8V6 44219884 IC50 = 8.3 nM T40016 C0R6PO 44220470 IC50 = 22 nM T40016 C0GW9R 44220471 IC50 = 16 nM T40016 C2ZV8C 44220675 IC50 = 20 nM T40016 CVF35J 44220676 IC50 = 8.5 nM T40016 CCR9E5 44220677 IC50 = 9.8 nM T40016 CU4Y0F 44222262 IC50 = 20 nM T40016 CR4O5D 44222437 IC50 = 16 nM T40016 CZHU72 44222438 IC50 = 12 nM T40016 CV6K2G 44222616 IC50 = 9.3 nM T40016 CXR5O7 44250279 IC50 = 62 nM T40016 C9QED8 44250280 IC50 = 17 nM T40016 CHGI03 44251606 IC50 = 13 nM T40016 C0OA6M 44264483 IC50 > 10000 nM T40016 COCE32 44264569 IC50 > 10000 nM T40016 CI0TN2 44264577 IC50 > 10000 nM T40016 CXOR54 44264579 IC50 > 10000 nM T40016 C01HSQ 44264588 IC50 > 10000 nM T40016 CP8OC7 44282950 Ki = 367 nM T40016 CT21MG 44292732 IC50 > 5000 nM T40016 CUS81V 44292816 IC50 = 310 nM T40016 CZ9MR4 44292832 IC50 = 40 nM T40016 C5QB1K 44292948 IC50 = 216.7 nM T40016 CBGI65 44293017 IC50 > 5000 nM T40016 CFR15U 44293099 IC50 = 310 nM T40016 CK8QL2 44293267 IC50 = 88 nM T40016 COF8L6 44293283 IC50 = 440 nM T40016 C9NO6K 44293320 IC50 = 15 nM T40016 C3LEM6 44293322 IC50 = 230 nM T40016 CMR51Y 44293351 IC50 = 23 nM T40016 C4C8ES 44293372 IC50 = 110 nM T40016 CJ6D4C 44294728 IC50 = 770 nM T40016 CJPD50 44294768 IC50 = 440 nM T40016 C6X2IH 44295653 Ki 10000 nM T40016 C1DBA2 44305237 IC50 = 324 nM T40016 CDB54J 44305270 IC50 = 177 nM T40016 C0XLN6 44305556 IC50 = 10 nM T40016 C17NWG 44305617 IC50 = 210 nM T40016 CHB82F 44305684 IC50 = 1929 nM T40016 C1UK4M 44305720 IC50 = 689 nM T40016 CTW67P 44305733 IC50 = 2170 nM T40016 CH4PU5 44305819 IC50 = 29 nM T40016 C7Y9TZ 44305822 IC50 = 31 nM T40016 CDXK57 44305874 IC50 = 3026 nM T40016 CP1MX9 44305909 IC50 = 1204 nM T40016 C6N1AR 44305929 IC50 = 1872 nM T40016 C9U6SZ 44306067 IC50 = 753 nM T40016 CE4S3K 44306078 IC50 = 812 nM T40016 C6OPD2 44306824 IC50 = 827 nM T40016 CLP97B 44310115 IC50 = 14000 nM T40016 C7F9NW 44310117 IC50 = 2700 nM T40016 CJ78FG 44310121 IC50 = 6600 nM T40016 CO7XP6 44310122 IC50 = 3800 nM T40016 CA73TS 44310248 IC50 = 25000 nM T40016 C2QV1X 44310288 IC50 = 220 nM T40016 CRT5J9 44310289 IC50 = 20 nM T40016 CD89XZ 44310345 IC50 = 1100 nM T40016 CKI2R0 44310353 IC50 = 1100 nM T40016 CQ17GY 44310359 IC50 = 2200 nM T40016 CKX52S 44310378 IC50 = 580 nM T40016 CD3X9U 44310397 IC50 = 850 nM T40016 CC2R3E 44310469 IC50 = 690 nM T40016 CMIG93 44310515 IC50 = 910 nM T40016 C7YKJ8 44310518 IC50 = 230 nM T40016 CV6AP0 44310535 IC50 = 42 nM T40016 C5A1XR 44310536 IC50 = 220 nM T40016 C7EWU8 44310595 IC50 = 130 nM T40016 CL42EC 44310626 IC50 = 110 nM T40016 CJH8Y1 44310641 IC50 = 570 nM T40016 CZ86HK 44310715 IC50 = 450 nM T40016 C4TU5G 44314208 IC50 = 16.7 nM T40016 CW21CA 44317747 Ki = 0.1 nM T40016 CT62WI 44341706 Ki = 394 nM T40016 CO10KF 44341745 Ki = 749 nM T40016 CP0AQ3 44341860 Ki = 130 nM T40016 CE62XL 44341871 Ki = 813 nM T40016 CIFK12 44341872 Ki = 158 nM T40016 C6KSD0 44341876 Ki = 51 nM T40016 CP6LV3 44341880 Ki = 533 nM T40016 C8RQS2 44342092 Ki = 260 nM T40016 CDGP02 44353994 IC50 = 188 nM T40016 C73CXK 44354006 Ki = 232 nM T40016 C0N3TD 44354884 IC50 = 900 nM T40016 CPQ2A6 44354885 Ki = 43 nM T40016 CM0G1V 44354886 IC50 = 780 nM T40016 CL6G3Q 44355066 IC50 = 35 nM T40016 C76OKZ 44370955 IC50 = 6.4 nM T40016 CZO25G 44371166 IC50 = 400 nM T40016 CILC83 44371259 IC50 = 1.4 nM T40016 CSAU31 44377064 IC50 > 10000 nM T40016 C7H9NC 44377081 IC50 > 10000 nM T40016 C60DYH 44377090 IC50 = 5800 nM T40016 CVH2R3 44377098 IC50 = 3000 nM T40016 CYLI63 44377110 IC50 > 10000 nM T40016 CQX39I 44377356 IC50 = 1400 nM T40016 C9FJW4 44377382 IC50 = 2100 nM T40016 C6SX0M 44393033 IC50 = 75 nM T40016 C7E9BC 44393047 IC50 = 460 nM T40016 CU4VI1 44393048 IC50 = 6.5 nM T40016 CM4DQ8 44393050 IC50 = 15 nM T40016 C2FJ0T 44393051 IC50 = 57 nM T40016 C8Y4RP 44393060 IC50 = 37 nM T40016 CK58MC 44393061 IC50 = 6.8 nM T40016 CTI0L9 44393062 IC50 = 23 nM T40016 CJ59US 44393181 IC50 = 71 nM T40016 CUK98X 44393182 IC50 = 170 nM T40016 C5NM4W 44393183 IC50 = 93 nM T40016 CFL1B2 44393188 IC50 > 1000 nM T40016 CMSV15 44393246 IC50 = 56 nM T40016 C12XBN 44393247 IC50 = 50 nM T40016 C89QJE 44394919 EC50 = 5.6 nM T40016 C5TY0K 44394965 IC50 = 165 nM T40016 C13SYV 44396250 Ki = 0.42 nM T40016 CB1P0S 44396251 Ki = 0.22 nM T40016 C0U5DZ 44396253 Ki = 0.16 nM T40016 CU3G0Y 44396254 Ki = 0.18 nM T40016 CHY1C3 44396271 Ki = 3 nM T40016 C29MBI 44396272 Ki = 2.1 nM T40016 C4TQ6N 44396282 Ki = 0.27 nM T40016 CH2Y3L 44396283 Ki = 0.27 nM T40016 CWZB52 44396284 Ki = 0.3 nM T40016 CD80LM 44396296 Ki = 0.4 nM T40016 C6SI5L 44396297 Ki = 0.39 nM T40016 CR4H1E 44396316 Ki = 0.42 nM T40016 C45LRH 44396317 Ki = 0.27 nM T40016 CPR85C 44396328 Ki = 0.22 nM T40016 CVF02B 44396329 Ki = 0.11 nM T40016 C5JG6H 44396330 Ki = 0.8 nM T40016 CA8V4G 44396331 Ki = 1.1 nM T40016 C57CPQ 44396332 Ki = 1.2 nM T40016 CGPV87 44396333 Ki = 6.5 nM T40016 CHG9O1 44396490 IC50 = 979 nM T40016 CPQL46 44396502 IC50 = 1812 nM T40016 CNH4C3 44396512 IC50 = 0.9 nM T40016 C1OYG3 44396526 IC50 = 870 nM T40016 CO25DV 44396547 IC50 = 1294 nM T40016 C7UP4O 44398565 IC50 = 5.012 nM T40016 CYCH34 44401707 IC50 = 9.1 nM T40016 CAG6T1 44401853 EC50 = 13 nM T40016 CA41SJ 44402030 IC50 = 10.2 nM T40016 C4PN2B 44402151 IC50 = 7.1 nM T40016 C61MGU 44402680 IC50 = 6.6 nM T40016 C9R8QP 44402681 IC50 = 8.5 nM T40016 CGL2T0 44402683 IC50 = 10 nM T40016 C63UET 44402699 IC50 = 8.4 nM T40016 C7VCZ5 44402711 IC50 = 7.1 nM T40016 CA5PI7 44402722 IC50 = 26 nM T40016 C2RLY1 44402736 IC50 = 2.2 nM T40016 CXI97U 44402746 IC50 = 8 nM T40016 C91WCI 44402753 IC50 = 5.6 nM T40016 CX4RZ6 44402754 IC50 = 5.5 nM T40016 C19KGF 44402755 IC50 = 18 nM T40016 CG4E3M 44402763 IC50 = 49 nM T40016 CRN9I4 44402766 IC50 = 10 nM T40016 C5Q6LX 44402767 IC50 = 3.1 nM T40016 CGRX27 44402769 IC50 = 24 nM T40016 C9R5SU 44402770 IC50 = 5.8 nM T40016 C7P6OT 44402796 IC50 = 10 nM T40016 C9XS4E 44402799 IC50 = 1.2 nM T40016 C1HE7G 44402805 IC50 = 2.1 nM T40016 CBUG70 44402817 IC50 = 2.7 nM T40016 CP1SY8 44402818 IC50 = 12 nM T40016 CBH76D 44402820 IC50 = 8.9 nM T40016 C7JU0O 44402832 IC50 = 21 nM T40016 CE5U1B 44402833 IC50 = 65 nM T40016 C36CWT 44402841 IC50 = 8.3 nM T40016 CW79UB 44402847 IC50 = 28 nM T40016 CP2IG4 44402961 IC50 > 2000 nM T40016 CXHF58 44403036 IC50 = 79 nM T40016 C25YCZ 44403037 IC50 > 2000 nM T40016 C6JNI4 44403038 EC50 = 2370 nM T40016 C45SOW 44403039 EC50 = 620 nM T40016 C1LUK3 44407314 IC50 = 2000 nM T40016 CA3B0O 44409475 Ki > 100 nM T40016 CYQZ19 44420005 IC50 = 481.5 nM T40016 CLA3J0 44420007 IC50 = 43 nM T40016 C1SFW5 44420010 IC50 = 0.7 nM T40016 C0C6FH 44420011 IC50 = 9 nM T40016 C0YG8R 44420014 IC50 = 0.4 nM T40016 CB1SU4 44420015 IC50 = 60.7 nM T40016 CHBG29 44420017 IC50 = 3.2 nM T40016 C5UIJ1 44420022 IC50 = 30.7 nM T40016 C91DUB 44420023 IC50 = 4.9 nM T40016 C2CJ6H 44420024 IC50 = 2.5 nM T40016 CAR8Y6 44420029 IC50 = 0.4 nM T40016 COD73E 44420033 IC50 = 1.5 nM T40016 CV38YP 44420040 IC50 = 0.7 nM T40016 CZFY86 44420051 IC50 = 1.5 nM T40016 C7I6RY 44420054 IC50 = 4.5 nM T40016 C5CW4E 44420057 IC50 = 0.1 nM T40016 CH1R7M 44420600 EC50 > 10 nM T40016 CF8N9J 44425531 IC50 = 204.3 nM T40016 CQ6R5N 44425537 IC50 = 33.4 nM T40016 CGY0M9 44425538 IC50 = 55.5 nM T40016 C6RGU2 44425539 IC50 = 166.9 nM T40016 CT7LE3 44425540 IC50 = 558 nM T40016 CT8Q9O 44425541 IC50 = 315 nM T40016 CE53FQ 44425542 IC50 > 3000 nM T40016 C0B6TU 44426753 Ki = 20 nM T40016 CO9JF7 44426754 Ki = 78 nM T40016 CV10KQ 44426759 Ki = 360 nM T40016 CF65BV 44426762 Ki = 470 nM T40016 CM01BZ 44426766 Ki = 19 nM T40016 C6EN4A 44426775 Ki = 154 nM T40016 CS5AL9 44426780 Ki = 227 nM T40016 CXZ4S3 44426781 Ki = 8.7 nM T40016 C8HO4K 44426782 Ki = 9.1 nM T40016 CXWC04 44426783 Ki = 31 nM T40016 C5OPU7 44426784 Ki = 14 nM T40016 CHT52I 44426787 Ki = 37 nM T40016 C35CJU 44426789 Ki = 45 nM T40016 C0FEN3 44426790 Ki = 7.1 nM T40016 CUK45W 44426792 Ki = 103 nM T40016 C19MJP 44426793 Ki = 4.9 nM T40016 CDN25Y 44426794 Ki = 46 nM T40016 C1ZDA4 44426795 Ki = 9.2 nM T40016 CFSH46 44426796 Ki = 6.5 nM T40016 CD0QH9 44426797 Ki = 47 nM T40016 C4FDY6 44427105 Ki = 4 nM T40016 C8OMK7 44427108 Ki = 1.8 nM T40016 C1M8YG 44427110 Ki = 0.9 nM T40016 CXO0S9 44427111 Ki = 0.6 nM T40016 C92VJT 44427112 Ki = 1.8 nM T40016 CY76PU 44427113 Ki = 4.8 nM T40016 C9AT0E 44427114 Ki = 2.7 nM T40016 CHMW84 44427115 Ki = 3 nM T40016 CM7TQ2 44427116 Ki = 31 nM T40016 C42FIO 44427117 Ki = 0.5 nM T40016 C79VAB 44427118 Ki = 1.1 nM T40016 CZM7N0 44430346 IC50 = 65.1 nM T40016 C2AJC1 44430347 IC50 = 64.8 nM T40016 C65HXP 44430353 IC50 = 62.7 nM T40016 C7O2JW 44430354 IC50 = 113.2 nM T40016 CK8QX3 44430355 IC50 = 51 nM T40016 CNB12D 44430370 IC50 = 56.6 nM T40016 CE36SB 44430377 IC50 = 48.9 nM T40016 CTS68I 44430382 IC50 = 36.3 nM T40016 C8BGC1 44430384 IC50 = 45.4 nM T40016 CI8JL5 44430385 IC50 = 43.5 nM T40016 CJ18XT 44430386 IC50 = 31.3 nM T40016 CG8KY9 44430387 IC50 = 22.1 nM T40016 CWR5Z1 44430388 IC50 = 80.3 nM T40016 CBST28 44430389 IC50 = 41.3 nM T40016 CUE9V4 44430390 IC50 = 65.8 nM T40016 C5CB2P 44430391 IC50 = 34.4 nM T40016 CV1DG2 44430392 IC50 = 175.3 nM T40016 C74CQT 44430393 IC50 = 341.6 nM T40016 CV6CM4 44430394 IC50 = 246.5 nM T40016 CEO60C 44430395 IC50 = 56 nM T40016 CVD9H1 44431137 IC50 > 10000 nM T40016 CD64XC 44431139 IC50 > 10000 nM T40016 C20KPU 44431142 IC50 = 1200 nM T40016 C12JEH 44431146 IC50 = 3600 nM T40016 CO4DF3 44431148 IC50 > 10000 nM T40016 C7ZDN6 44431150 IC50 = 1900 nM T40016 C3WSV5 44431167 IC50 = 1300 nM T40016 CXW14R 44431168 IC50 > 2000 nM T40016 CJR34C 44431169 IC50 > 2000 nM T40016 CP6L8E 44431172 IC50 > 2000 nM T40016 CIOW01 44431179 IC50 > 2000 nM T40016 CECG82 44431181 IC50 > 2000 nM T40016 C06NTR 44431183 IC50 > 2000 nM T40016 CQXD51 44431187 IC50 = 490 nM T40016 CLJC40 44431190 IC50 = 120 nM T40016 CL1XK9 44431202 IC50 = 79 nM T40016 C7VGK1 44433485 IC50 < 1000 nM T40016 C3E2QI 44433486 IC50 = 30.2 nM T40016 CK6P9M 44433489 IC50 = 7.586 nM T40016 CV4I9Z 44433491 IC50 = 5.888 nM T40016 C2R5SU 44433492 IC50 = 3.631 nM T40016 C4DFA6 44433500 IC50 = 4.677 nM T40016 C7IYB1 44433501 IC50 = 8.511 nM T40016 CR3OW8 44433502 IC50 = 3.715 nM T40016 C1Z0QH 44433503 EC50 = 1.202 nM T40016 C3SJ5V 44433504 Ki = 387 nM T40016 C2SCP7 44435606 IC50 > 1600 nM T40016 CH5E3L 44435611 IC50 > 1300 nM T40016 CDO62N 44435656 IC50 = 20 nM T40016 C9TP4C 44435662 IC50 = 19 nM T40016 C19TMW 44435663 IC50 = 27 nM T40016 C90WUC 44435667 IC50 = 21 nM T40016 CHFB89 44435668 IC50 = 11 nM T40016 C8IWK2 44435669 IC50 = 8 nM T40016 C8SG5B 44441950 Ki = 10 nM T40016 CWKU75 44441951 Ki = 10 nM T40016 C9EG5T 44441952 Ki = 3 nM T40016 CV0UD9 44441953 Ki = 9 nM T40016 C1OCJ7 44441954 IC50 = 10 nM T40016 CWH06J 44441955 Ki = 20 nM T40016 C9IS3X 44441956 Ki = 56.3 nM T40016 CJQ5G8 44441958 Ki > 3000 nM T40016 CU32PK 44441961 Ki = 59.8 nM T40016 CJ5E0V 44441962 Ki > 3000 nM T40016 C60DXZ 44442904 Ki > 10000 nM T40016 CIM40U 44442905 Ki > 10000 nM T40016 C8PIL1 44442906 Ki > 10000 nM T40016 CB3QN1 44442907 Ki > 10000 nM T40016 CY7UK6 44442908 Ki = 1200 nM T40016 CFX0E8 44442909 Ki > 5000 nM T40016 CV3S1P 44442910 Ki = 3700 nM T40016 C8KDU3 44442911 Ki > 10000 nM T40016 CW8CZ2 44442912 Ki = 1000 nM T40016 CTUE70 44442913 Ki = 4450 nM T40016 CA48OP 44442916 Ki = 3000 nM T40016 CXHK75 44442917 Ki = 1250 nM T40016 CL6ZK2 44442918 Ki = 800 nM T40016 C7YH5D 44442919 Ki = 196 nM T40016 CL7H0E 44442920 Ki = 216 nM T40016 CF7GX1 44442921 Ki = 1300 nM T40016 CMN07E 44442922 Ki > 10000 nM T40016 CJ3L7N 44442923 Ki = 163 nM T40016 CV4L6Z 44442924 Ki = 432 nM T40016 CT3B8Y 44442925 Ki = 193 nM T40016 CEQN26 44442926 Ki = 99 nM T40016 C7ZV0W 44442927 Ki = 4 nM T40016 C9E2QR 44442928 Ki > 10000 nM T40016 CO70RC 44442929 Ki = 55 nM T40016 C96ZLT 44442930 Ki = 1950 nM T40016 CE32IH 44442932 Ki = 2100 nM T40016 CG1VI4 44442933 Ki = 950 nM T40016 CFX2Z6 44442935 Ki = 137 nM T40016 C8JSW1 44442936 Ki = 750 nM T40016 CVQ5K4 44442937 Ki = 113 nM T40016 CIJ9N6 44442938 Ki = 64 nM T40016 CFM0Y1 44442939 IC50 = 3200 nM T40016 C31QCR 44442951 Ki = 76 nM T40016 CQGR94 44442953 Ki = 6 nM T40016 CNBU39 44442955 Ki = 4 nM T40016 C9LT3P 44442957 Ki = 5 nM T40016 C8PE5X 44442960 Ki = 9 nM T40016 C1GL4Z 44442962 Ki = 45 nM T40016 CK4YB1 44442964 Ki = 65 nM T40016 CHC51X 44442967 Ki = 99 nM T40016 CI37JQ 44442979 Ki = 15 nM T40016 C3RUQ9 44442980 Ki = 13 nM T40016 CZL8H0 44442982 Ki = 56 nM T40016 C8S1OM 44442983 Ki = 13 nM T40016 CQX76V 44442984 Ki = 2 nM T40016 COE4T0 44442986 Ki = 9 nM T40016 CY7M3O 44442988 Ki = 10 nM T40016 CMV0G6 44443285 IC50 = 210 nM T40016 CM2JI8 44443286 IC50 = 460 nM T40016 CAS57C 44443287 IC50 = 14000 nM T40016 CQY8H1 44443288 IC50 = 23 nM T40016 C4NQ1C 44443289 IC50 = 82 nM T40016 C0WMP8 44443290 IC50 = 540 nM T40016 CQ0N2S 44443291 IC50 > 10000 nM T40016 CW30DO 44443292 IC50 = 660 nM T40016 CH7B1G 44454500 Ki = 3.8 nM T40016 CDEP04 44454503 Ki = 1.4 nM T40016 CJY2X9 44454504 Ki = 1.2 nM T40016 C94YHC 44454533 Ki = 1 nM T40016 C1YSC6 44454535 Ki = 1.5 nM T40016 C3IW0D 44454537 Ki = 2.3 nM T40016 C9L5XM 44454539 Ki = 1.3 nM T40016 C48ZEN 44454540 Ki = 2.2 nM T40016 C2BQ0E 44454565 Ki = 1.7 nM T40016 CY78VG 44454566 Ki = 1.2 nM T40016 C2LJ6Q 44454567 Ki = 22 nM T40016 C30CHA 44454624 Ki = 2.1 nM T40016 CU7F5L 44454647 Ki = 2.4 nM T40016 CY7NS9 44454672 Ki = 0.8 nM T40016 CAT25W 44454673 Ki > 1000 nM T40016 CEFI01 44454699 Ki = 0.8 nM T40016 C41YOI 44454723 Ki = 0.5 nM T40016 C4ZVS8 44454724 Ki = 0.3 nM T40016 CEI8J6 44454725 Ki = 0.9 nM T40016 C0MG5R 44454751 Ki = 0.8 nM T40016 C49BKG 44454777 Ki = 0.8 nM T40016 C8KXU2 44454778 Ki = 0.5 nM T40016 C6S8ZH 44454802 Ki = 6.7 nM T40016 CC42DA 44454804 Ki = 1 nM T40016 CMB16K 44454805 Ki = 0.9 nM T40016 CE0Y5C 44454806 Ki = 1.6 nM T40016 CCU20Z 44454807 Ki = 8.6 nM T40016 CSV3G4 44454832 Ki = 1.6 nM T40016 CHX6B1 44454869 Ki = 1.1 nM T40016 CB5G1W 44454870 Ki = 3.4 nM T40016 CZ37QB 44454903 Ki = 1.5 nM T40016 CM6LE3 44454906 Ki = 3.7 nM T40016 CCB2O8 44454938 Ki = 9 nM T40016 CKXH14 44454942 Ki = 34 nM T40016 CYG7X4 44473146 IC50 = 0.062 nM T40016 CR5SI0 44476535 EC50 > 10000 nM T40016 C0B2ZT 44515373 IC50 = 0.032 nM T40016 C0MVJ3 44516035 IC50 = 0.051 nM T40016 CM29JD 44516036 IC50 = 1 nM T40016 CKHJ76 44517735 IC50 = 0.3162 nM T40016 CR19IH 44543858 IC50 = 180 nM T40016 C05HEP 44543860 IC50 = 45 nM T40016 C45ZHO 44543969 IC50 = 120 nM T40016 C27TZY 44543970 IC50 = 19 nM T40016 C25OXZ 44544094 IC50 = 370 nM T40016 C7JIF6 44544321 IC50 = 40 nM T40016 C1M4BL 44544711 IC50 = 2.4 nM T40016 CK1Z8P 44545482 IC50 = 43 nM T40016 CF6V4G 44563171 EC50 = 1.995 nM T40016 CSN41Q 44563745 EC50 = 2500 nM T40016 CP6F3O 44563746 EC50 = 33 nM T40016 C46TRW 44563747 EC50 = 1860 nM T40016 C80WGP 44565589 EC50 = 1067.3 nM T40016 CU40ER 44565590 EC50 = 1159.6 nM T40016 CJ39EH 44565614 EC50 = 678.1 nM T40016 C6WO3E 44565615 EC50 = 9.9 nM T40016 CQZ78D 44565616 EC50 = 12.3 nM T40016 CFZD18 44565646 Ki = 5.4 nM T40016 CK8MH3 44565647 Ki = 0.9 nM T40016 CEZ35O 44565648 Ki = 37.8 nM T40016 C6Q5DK 44569945 EC50 = 1.995 nM T40016 C8S3RZ 44570143 EC50 = 25.12 nM T40016 CD65UK 44570182 EC50 = 50.12 nM T40016 C14JOH 44570183 EC50 = 794.33 nM T40016 C06LMN 44570222 EC50 = 3.162 nM T40016 CK10JY 44570223 IC50 = 398.11 nM T40016 CBET53 44570224 EC50 = 251.19 nM T40016 C9TVI8 44570225 EC50 = 25.12 nM T40016 CVO8L1 44570275 EC50 = 50.12 nM T40016 C8BGL6 44585565 IC50 = 1300 nM T40016 C93AMI 44586093 IC50 = 36 nM T40016 CS81IL 44587000 IC50 = 3.6 nM T40016 CUNV59 44587001 IC50 = 2.8 nM T40016 CMN58Z 44587002 IC50 = 2.1 nM T40016 C9RX7K 44587056 IC50 = 21.5 nM T40016 C71CKD 44587057 IC50 = 17.4 nM T40016 C7LU9Z 44587058 IC50 = 2.4 nM T40016 CCJ6Z0 44587059 IC50 = 28.6 nM T40016 C68ZVD 44587197 IC50 = 0.5 nM T40016 CF93RA 44587198 IC50 = 55.1 nM T40016 CIHA86 44587199 IC50 = 352 nM T40016 C68JWV 44587218 IC50 = 12.3 nM T40016 C2USW6 44587219 IC50 = 5.7 nM T40016 CDBQ16 44587220 IC50 = 3.8 nM T40016 CUA45E 44587248 IC50 = 3.5 nM T40016 CC0V2T 44587249 IC50 = 5.8 nM T40016 COU07A 44587250 IC50 = 5.2 nM T40016 C91YAW 44587251 IC50 = 1.3 nM T40016 CJ3VI8 44593465 Ki = 1.3 nM T40016 C70MSI 44593549 EC50 = 158.49 nM T40016 CL8O7P 44769019 IC50 > 6309.57 nM T40016 C9PLK4 45263610 IC50 = 110 nM T40016 C78JKD 45265930 IC50 = 40 nM T40016 C1Z9XI 45267345 IC50 = 1400 nM T40016 CWKP29 45267349 IC50 = 150 nM T40016 CN8HI2 45267356 IC50 > 3000 nM T40016 CG6X9E 45267360 IC50 = 41 nM T40016 CJ10QV 45267605 IC50 = 0.7943 nM T40016 C3KD4Q 45267606 IC50 = 0.3981 nM T40016 CGN7S5 45267615 IC50 = 0.1995 nM T40016 CK04FJ 45267900 IC50 = 460 nM T40016 CPB29I 45268475 IC50 = 31.62 nM T40016 CV7JG9 45268476 IC50 = 25.12 nM T40016 CK0W2Z 45268480 IC50 = 7.943 nM T40016 CF0N2I 45268481 IC50 = 2.512 nM T40016 CF9B0L 45268482 IC50 = 5.012 nM T40016 CQ1F4T 45268485 IC50 = 0.3981 nM T40016 CX7ZG0 45268785 IC50 = 14 nM T40016 CD7T3W 45269091 IC50 = 68 nM T40016 C93BLG 45269348 IC50 = 0.2512 nM T40016 CJTC89 45269354 IC50 = 0.2512 nM T40016 CLSH89 45269632 IC50 = 23 nM T40016 CD61HS 45269633 IC50 = 5.7 nM T40016 CGIT19 45269634 IC50 = 550 nM T40016 C21HYG 45269951 IC50 = 7 nM T40016 CAP56V 45269952 IC50 = 110 nM T40016 CKG49L 45269958 IC50 = 21 nM T40016 C9FK5M 45270463 IC50 = 21 nM T40016 C8ICF3 45270464 IC50 = 480 nM T40016 CIR20D 45270774 IC50 = 20 nM T40016 C9D1IT 45270779 IC50 = 58 nM T40016 C6HZ3T 45271025 IC50 = 0.5012 nM T40016 CS6LO7 45271294 IC50 = 15 nM T40016 CS26QV 45271295 IC50 = 27 nM T40016 C1S8IW 45271296 IC50 = 26 nM T40016 C8GSB6 45271297 IC50 = 840 nM T40016 CJKN81 45271616 IC50 = 132 nM T40016 C08UBE 45272032 IC50 > 10000 nM T40016 C9MF3P 45272514 IC50 = 26 nM T40016 CBEC80 45273046 IC50 = 14 nM T40016 CT52NO 45273047 IC50 = 21 nM T40016 CZXN64 45273048 IC50 = 34 nM T40016 CUZ5C6 45273374 IC50 = 102 nM T40016 C4LK8X 45273665 IC50 = 3.162 nM T40016 CQ81DI 45273670 IC50 = 0.3162 nM T40016 CR8I9S 45486375 Ki = 2 nM T40016 CP35QW 45486376 Ki = 47 nM T40016 C4XDQ1 45486377 Ki = 11 nM T40016 CAT4C2 45486382 Ki = 7 nM T40016 CDA24N 45486383 Ki = 1 nM T40016 C9YM2G 45486384 Ki = 2 nM T40016 CX8HO5 45486385 Ki = 2.6 nM T40016 CJX89Y 45486393 EC50 = 2 nM T40016 C8K2DM 45486403 Ki = 2 nM T40016 CQT1C9 45486404 Ki = 5.2 nM T40016 C0RID5 45486424 Ki = 2.5 nM T40016 C0WQ4R 45486436 Ki = 21 nM T40016 COG73H 45486437 Ki = 2 nM T40016 C2NWO7 45486438 Ki = 2 nM T40016 CM8F4H 45486439 Ki = 9 nM T40016 CD7L1N 45486442 Ki = 8 nM T40016 CW20GE 45486443 Ki = 1 nM T40016 C5HL9V 45486450 Ki = 1.5 nM T40016 CW7J5K 45486451 Ki = 4 nM T40016 CJ6LH2 45486455 EC50 = 1.8 nM T40016 CL91NK 45486456 Ki = 2.5 nM T40016 C6OYN8 45486457 Ki = 1 nM T40016 C3KU7H 45486464 Ki = 3 nM T40016 C14DQK 45486465 Ki = 31 nM T40016 CR6P7Z 45486470 Ki = 3.9 nM T40016 CU3IY5 45486473 Ki = 2 nM T40016 CHRX37 45486474 Ki = 4.3 nM T40016 CY54HC 45486477 Ki = 2 nM T40016 CX8LZ0 45486478 Ki = 7.9 nM T40016 C7PMW0 45486484 Ki = 33 nM T40016 COD9R1 45486485 Ki = 2 nM T40016 CLT46H 45789439 Ki = 18 nM T40016 C1BYW8 46830503 IC50 = 3162.28 nM T40016 C04BWG 46830504 IC50 = 251.19 nM T40016 CY2ZJ0 46830505 IC50 = 3162.28 nM T40016 CC45TP 46830506 IC50 > 10000 nM T40016 CN7Q8A 46830507 IC50 = 398.11 nM T40016 C0QT3G 46830795 IC50 > 2511.89 nM T40016 C0JCX3 46830796 IC50 > 10000 nM T40016 CMS6R9 46830797 IC50 = 1258.93 nM T40016 CJIN74 46830798 IC50 = 3162.28 nM T40016 CRY31M 46830799 IC50 > 10000 nM T40016 CKA07I 46830800 IC50 = 501.19 nM T40016 C4XRF9 46830801 IC50 = 2511.89 nM T40016 C2NC3V 46831087 IC50 = 630.96 nM T40016 CXP6K3 46831397 IC50 = 794.33 nM T40016 C0QNC9 46831400 IC50 = 1258.93 nM T40016 CX6L7Q 46831696 IC50 = 19.95 nM T40016 CQ1IP3 46831697 IC50 = 1995.26 nM T40016 CL1KR4 46831698 IC50 = 31.62 nM T40016 C1DH9W 46831699 IC50 = 39.81 nM T40016 CASV14 46831700 IC50 = 1995.26 nM T40016 CTXY26 46831701 IC50 = 1584.89 nM T40016 CG0J5K 46831956 IC50 = 3162.28 nM T40016 CY3WK4 46831957 IC50 = 1995.26 nM T40016 CP19UN 46831958 IC50 = 15.85 nM T40016 CBJZ85 46831959 IC50 = 50.12 nM T40016 CE4VC8 46831960 IC50 = 251.19 nM T40016 CAR23U 46832233 IC50 = 125.89 nM T40016 CUAO43 46832234 EC50 = 316.23 nM T40016 CM40EP 46832235 IC50 = 15.85 nM T40016 CJ32XT 46832236 IC50 = 25.12 nM T40016 C81GUN 46832237 IC50 = 50.12 nM T40016 CT31AL 46832511 IC50 = 12.59 nM T40016 CR15XE 46832512 IC50 = 39.81 nM T40016 CW12GM 46832513 IC50 = 15.85 nM T40016 C0GTK8 46832514 EC50 = 199.53 nM T40016 C8HO0L 46832515 IC50 = 100 nM T40016 C2S6PL 46834818 IC50 > 10000 nM T40016 C9F5OB 46883794 IC50 = 63.1 nM T40016 C60NSG 46883795 IC50 = 63.1 nM T40016 CHNI89 46883838 IC50 = 158.49 nM T40016 C7KW8T 46883839 IC50 = 199.53 nM T40016 CM7EA1 46883840 IC50 = 199.53 nM T40016 C06JMN 46883842 IC50 = 251.19 nM T40016 CZSG25 46883893 IC50 = 251.19 nM T40016 CQD4K2 46883894 IC50 = 398.11 nM T40016 CMA7J9 46883895 IC50 = 398.11 nM T40016 CBY2M8 46883896 IC50 = 1000 nM T40016 CZDB52 46883897 IC50 > 6309.57 nM T40016 CZI1H6 46883898 IC50 > 6309.57 nM T40016 CV34LD 46883930 IC50 > 6309.57 nM T40016 CJ7TW5 46883931 IC50 > 6309.57 nM T40016 CTE7B2 46883932 IC50 > 6309.57 nM T40016 CAIF17 46883933 IC50 > 6309.57 nM T40016 CA9D4X 46883934 IC50 = 251.19 nM T40016 CXNT91 46883998 IC50 = 251.19 nM T40016 CCH3B0 46883999 IC50 = 251.19 nM T40016 CGSD50 46884000 IC50 = 316.23 nM T40016 C4VKF7 46884001 IC50 = 316.23 nM T40016 CHV9D6 46884030 IC50 = 501.19 nM T40016 CHW0T8 46884031 IC50 = 794.33 nM T40016 C68YXV 46884032 IC50 > 6309.57 nM T40016 CYB42R 46885327 Ki = 51 nM T40016 CA64WN 46885370 Ki = 6.9 nM T40016 C3S2EW 46885371 Ki = 18 nM T40016 CVD89I 46885372 Ki = 4.2 nM T40016 C1NX3S 46885418 Ki = 30 nM T40016 CXQ19B 46885419 Ki = 2465 nM T40016 C2X0TL 46885420 Ki = 3210 nM T40016 C3SB4Y 46885484 Ki = 4109 nM T40016 CNG65D 46888392 IC50 = 10000 nM T40016 C2WQ4M 46888393 IC50 = 2113 nM T40016 CTEY73 46888414 IC50 = 2089 nM T40016 C82NDU 46888415 IC50 = 178 nM T40016 CF97JD 46888416 IC50 = 52 nM T40016 CI4HJ9 46888439 IC50 = 72 nM T40016 CI6Q5G 46888440 IC50 = 99 nM T40016 CAE10V 46888443 IC50 = 30 nM T40016 C1N4WH 46888464 IC50 = 282 nM T40016 C5L7NY 46888465 IC50 = 54 nM T40016 CJK47T 46888466 IC50 = 35 nM T40016 C9QO6J 46888468 IC50 = 14 nM T40016 C6DB3K 46888487 EC50 = 93 nM T40016 C72MUY 46889765 IC50 > 5000 nM T40016 C6DVO1 46889848 IC50 > 10000 nM T40016 CZ90FC 46894119 IC50 > 25000 nM T40016 C3Q7RI 46913890 IC50 > 10000 nM T40016 CP91XE 46914741 IC50 > 10000 nM T40016 CTM2J5 46915203 IC50 > 10000 nM T40016 C75IFZ 46915353 IC50 > 10000 nM T40016 CX70GY 46915355 IC50 > 10000 nM T40016 C7NC4B 46917090 IC50 > 10000 nM T40016 C2LCJ7 46937290 IC50 = 3.3 nM T40016 CKQ8J3 46937431 IC50 = 8 nM T40016 CL7P3N 46938234 IC50 > 9497 nM T40016 CFJT93 46938236 IC50 = 6800 nM T40016 C8P7JH 46938914 IC50 = 860 nM T40016 CY95VK 46938915 IC50 = 690 nM T40016 CVX25Q 46938916 IC50 = 3 nM T40016 C2V5AT 46939019 IC50 = 12 nM T40016 C5R6GI 46939020 IC50 = 8 nM T40016 CF1BX0 46939115 IC50 = 27 nM T40016 C4P0EU 46939116 IC50 = 11 nM T40016 CD6B7X 46939395 IC50 = 1.4 nM T40016 C1KXF2 46939396 IC50 = 1700 nM T40016 CVRU79 46943298 Ki = 2.5 nM T40016 C4Z3NF 49652111 EC50 = 109500 nM T40016 CTG0U1 49652409 EC50 = 109000 nM T40016 CX0NO8 49782554 IC50 < 15848.93 nM T40016 CC7T8Q 49782555 EC50 < 15848.93 nM T40016 CD07EV 49782777 EC50 < 15848.93 nM T40016 C43UKW 49782778 IC50 < 9246.98 nM T40016 C2JTF0 49782779 EC50 < 15848.93 nM T40016 CS7KX9 49782780 EC50 < 15848.93 nM T40016 C36RYU 49782781 IC50 < 13489.63 nM T40016 C8OA0C 49782985 EC50 < 15848.93 nM T40016 C5Y6QU 49782986 IC50 = 3126.08 nM T40016 CB8V7R 49782987 EC50 < 15848.93 nM T40016 CU3S6H 49836028 Ki = 0.7 nM T40016 C96SLW 49851364 Ki = 1.2 nM T40016 C54IGW 49851365 Ki = 18.7 nM T40016 C0G1UO 49851366 Ki = 0.6 nM T40016 CN57XD 49851367 Ki = 20.7 nM T40016 CO5XW9 49851368 Ki = 4.6 nM T40016 CDN4K6 49851369 Ki = 0.4 nM T40016 C0K7OD 49851464 Ki = 0.9 nM T40016 C2JU6O 49851465 Ki = 7.3 nM T40016 CIO2F8 49851466 Ki = 1.1 nM T40016 C4YXN1 49851467 Ki = 0.7 nM T40016 C16OCR 49851468 Ki = 0.4 nM T40016 CI0MX2 49851469 Ki = 2.2 nM T40016 CA4UP7 49851577 Ki = 58.7 nM T40016 CFN03Q 49851580 Ki = 5.7 nM T40016 CUD91T 49862248 EC50 > 10000 nM T40016 CTKV39 49864176 IC50 > 10000 nM T40016 CHT86O 50925620 EC50 = 7300 nM T40016 CCM1T9 50938547 IC50 = 7.943 nM T40016 CZ8J1V 50942115 Ki = 1.7 nM T40016 C23OEF 50942312 EC50 = 12.59 nM T40016 CTHL29 50993207 EC50 = 5600 nM T40016 CH2M5E 50993208 EC50 = 50800 nM T40016 CC54NG 50993209 EC50 = 25300 nM T40016 CM2BI1 50993282 EC50 = 123500 nM T40016 C6DIX2 50993355 EC50 = 101000 nM T40016 CX1KO8 51346768 Ki = 523 nM T40016 C7N9TD 51346823 EC50 = 0.6 nM T40016 C0WDX3 51347001 Ki = 2.9 nM T40016 CF8DK7 51347002 Ki = 9.4 nM T40016 CTH45Q 52918523 IC50 = 0.17 nM T40016 CEC4I7 52941608 IC50 = 23 nM T40016 C6NR7I 52942081 EC50 > 10000 nM T40016 CDV90J 52942528 IC50 = 15.85 nM T40016 CZ1DS4 52943487 EC50 = 130000 nM T40016 C8Y9SU 52944898 IC50 > 1000 nM T40016 CTV7K1 53316621 EC50 = 5.012 nM T40016 CLC5U1 53316851 EC50 = 25.12 nM T40016 C82ATJ 53316852 EC50 = 25.12 nM T40016 C0YNS6 53317029 Ki = 2.3 nM T40016 C0KZW5 53317030 Ki = 2.4 nM T40016 CVNU71 53317031 Ki = 5 nM T40016 CY61KR 53317043 IC50 = 0.1995 nM T40016 C6EZS2 53317044 IC50 = 15.85 nM T40016 CO5GV1 53317045 IC50 = 5.012 nM T40016 CK5UT4 53317489 Ki = 157 nM T40016 CSY4T6 53317533 IC50 = 1.259 nM T40016 CB38MW 53317966 IC50 = 0.1259 nM T40016 C9Y0RM 53318166 EC50 = 10 nM T40016 CCT76B 53318167 EC50 = 12.59 nM T40016 CQ8K1O 53318317 Ki = 38.3 nM T40016 CO7Q4T 53318326 IC50 = 125.89 nM T40016 CQI41V 53318658 Ki = 436 nM T40016 CM0LU1 53318659 Ki = 10 nM T40016 CQBZ97 53318680 EC50 = 15 nM T40016 CAWQ20 53319309 IC50 = 12.59 nM T40016 CC8KA2 53319310 IC50 = 31.62 nM T40016 CPS1C0 53319665 EC50 = 5.7 nM T40016 CVIE23 53319666 Ki = 1.8 nM T40016 CUD48O 53320087 Ki = 6.39 nM T40016 C2CS5A 53320355 Ki = 2.2 nM T40016 C2DM5A 53320607 IC50 = 5.012 nM T40016 C4J1DL 53320608 IC50 = 63.1 nM T40016 C7Z0PN 53320971 IC50 = 3.8 nM T40016 C05MAE 53320972 Ki = 3.5 nM T40016 C58WMJ 53321241 Ki = 3 nM T40016 C5ITY0 53321440 IC50 = 6.31 nM T40016 C0US8P 53321674 IC50 = 7.943 nM T40016 CD2NZ1 53321685 IC50 = 5.7 nM T40016 CB67IZ 53321912 IC50 = 0.07943 nM T40016 CP9FI6 53321913 IC50 = 7.943 nM T40016 C7VWT1 53322135 EC50 = 31.62 nM T40016 C8ZB5U 53322300 EC50 = 0.9 nM T40016 CD2AW1 53322301 Ki = 11.7 nM T40016 CHQ5A9 53322303 Ki = 1.3 nM T40016 CO4ZQ2 53322313 IC50 = 0.2512 nM T40016 C97KUE 53322314 IC50 = 1.995 nM T40016 C63BYE 53322904 IC50 = 19.95 nM T40016 CDL2K7 53323256 IC50 = 3.981 nM T40016 CIQ28P 53323257 IC50 = 50.12 nM T40016 C4MJ9W 53323258 IC50 = 5.012 nM T40016 C4X3VU 53323259 IC50 = 1.995 nM T40016 CJD29K 53323475 EC50 = 3.981 nM T40016 CD0N1K 53323476 EC50 = 1000 nM T40016 CQ41DA 53323656 Ki = 9 nM T40016 C4I3OP 53323657 Ki = 0.9 nM T40016 CH8LW2 53323658 Ki = 106 nM T40016 CKRC57 53323670 IC50 = 0.3162 nM T40016 C9G2SP 53323671 IC50 = 5.012 nM T40016 CBM23P 53323672 IC50 = 50.12 nM T40016 C7K9RF 53323962 EC50 = 5.1 nM T40016 C4WC2R 53324599 IC50 = 7.943 nM T40016 C8EM1C 53324945 Ki = 3.1 nM T40016 CH2U4P 53324954 IC50 = 125.89 nM T40016 C16TGD 53325224 Ki = 416 nM T40016 CK2BN3 53325565 Ki = 10.4 nM T40016 CIU8H2 53325583 EC50 = 12.59 nM T40016 CLG69E 53325612 EC50 = 1.995 nM T40016 CYH3V0 53325642 Ki = 50.2 nM T40016 CP7Y9M 53326069 EC50 = 6.31 nM T40016 C7Q8CZ 53326228 EC50 = 0.4 nM T40016 CPFW50 53326229 EC50 = 0.2 nM T40016 C02REC 53326230 Ki = 19.6 nM T40016 C1Z0MJ 53326231 Ki = 8 nM T40016 C79XKL 53326232 Ki = 1 nM T40016 CXJ84N 53326233 Ki = 157 nM T40016 C68EWU 53326245 IC50 = 39.81 nM T40016 CTX3I2 53326246 IC50 = 3.162 nM T40016 CGX19M 53326247 IC50 = 794.33 nM T40016 C9HN7W 53326537 Ki = 132 nM T40016 CB71TJ 53326538 Ki = 12.2 nM T40016 C82DYI 53326614 Ki > 4290 nM T40016 C6K2OB 53328064 Ki = 0.66 nM T40016 CJCP75 53359074 Ki = 1.64 nM T40016 C9H5YE 53361128 EC50 > 10000 nM T40016 C9XT0F 53483966 EC50 = 2.97 nM T40016 CUR24K 53875787 IC50 = 340 nM T40016 C30XLO 54592009 IC50 = 597 nM T40016 CCJ42Y 56589543 IC50 = 3540 nM T40016 CW9OS3 56593697 Ki = 49.5 nM T40016 CU02PM 56593698 Ki = 1.2 nM T40016 CUX1B9 56593851 Ki = 3.8 nM T40016 CJ98FM 56593852 Ki = 4 nM T40016 CN0Q8R 56593853 Ki = 2.9 nM T40016 CEN7V4 56593854 Ki = 3.9 nM T40016 C1YGH6 56593980 Ki = 6 nM T40016 CV0JW2 56593981 Ki = 2.5 nM T40016 C8G0AR 56593982 Ki = 9.17 nM T40016 C47DRS 56593983 Ki = 5.48 nM T40016 C9W5DZ 56593984 Ki = 1.74 nM T40016 CV9OE8 56594117 Ki = 486 nM T40016 CA9ER8 56594118 Ki = 1.6 nM T40016 CXQ2R5 56594120 Ki = 1.3 nM T40016 C7ULR4 56594121 Ki = 1.68 nM T40016 C6ZR3U 56594268 Ki = 2.6 nM T40016 CKB34M 56594269 Ki = 2.7 nM T40016 C4P7JM 56594270 Ki = 1.96 nM T40016 CNOI17 56594271 Ki = 2.53 nM T40016 C42NTL 56594272 Ki = 3.08 nM T40016 CO0CR2 56594389 Ki = 8.6 nM T40016 CY0ZX3 56594392 Ki = 4.1 nM T40016 C7UVE6 56594518 Ki = 4.2 nM T40016 CH0M6A 56594523 Ki = 15.4 nM T40016 CR4U9K 56594613 IC50 = 4960 nM T40016 CV39IP 56595706 Ki = 7.1 nM T40016 CTSJ36 56595707 Ki = 10.5 nM T40016 C7KU1Y 56595708 Ki = 24 nM T40016 CEY96L 56595709 Ki = 2.5 nM T40016 CI1UN4 56661440 EC50 = 0.43 nM T40016 C1L0FO 56664884 EC50 = 0.38 nM T40016 CU5C3L 56668302 EC50 = 8.78 nM T40016 CI2E4M 56671781 EC50 = 0.71 nM T40016 CX5LM7 56671782 EC50 = 3.93 nM T40016 C4F7OS 56671783 EC50 = 7.35 nM T40016 CKHZ50 56675193 EC50 = 1.87 nM T40016 CUM21Y 56677234 Ki = 2.9 nM T40016 CBG79E 56681836 EC50 = 0.78 nM T40016 CR3P4L 56681837 EC50 = 1.75 nM T40016 CR4IK7 56681838 EC50 = 2.82 nM T40016 CF3G2M 56925477 IC50 = 3500 nM T40016 CZ7O8G 56925478 IC50 = 950 nM T40016 CW87RG 56925573 IC50 > 10000 nM T40016 C30DAL 56925669 IC50 = 5500 nM T40016 CQHA65 56925670 IC50 > 10000 nM T40016 CJP31U 56925671 IC50 > 10000 nM T40016 CI3S6F 56925790 IC50 > 10000 nM T40016 CTY1Q9 56925791 IC50 = 6900 nM T40016 CTG9I7 56926011 IC50 = 200 nM T40016 CL16UQ 56949326 IC50 < 10000 nM T40016 CX6Q9M 57390301 Ki = 1.6 nM T40016 CR3Y4C 57390331 IC50 = 1.4 nM T40016 C2PAW0 57390332 IC50 = 14.3 nM T40016 C26UES 57390369 EC50 = 22.4 nM T40016 C3Y9SF 57390753 IC50 = 61 nM T40016 C7R4HE 57390754 IC50 = 60 nM T40016 CM0SG2 57390990 IC50 = 87 nM T40016 CD1KG0 57391329 IC50 = 17.6 nM T40016 C1ETU3 57391330 IC50 = 23.5 nM T40016 C5Q0AF 57392164 IC50 = 2.1 nM T40016 C4SD8X 57392560 IC50 = 13 nM T40016 CU8AN3 57392780 IC50 = 88 nM T40016 CX12JM 57392781 IC50 = 3 nM T40016 C9OMW1 57392782 IC50 = 405 nM T40016 C6YQU8 57393091 IC50 = 17.2 nM T40016 C8BPN6 57393863 IC50 = 2.85 nM T40016 CS50GQ 57393864 IC50 = 9.7 nM T40016 C8S0HJ 57394288 IC50 = 23 nM T40016 C30JOV 57394501 IC50 = 7 nM T40016 C76QKN 57394818 IC50 = 70.2 nM T40016 CY6H7M 57394819 IC50 = 118 nM T40016 C8N0BF 57394833 IC50 = 722 nM T40016 CF8H1A 57394834 IC50 = 5.1 nM T40016 CDJ67U 57395566 Ki = 1 nM T40016 CW5V3Q 57395588 IC50 = 3.8 nM T40016 CM5UX2 57395589 IC50 = 2.2 nM T40016 CST3E8 57395590 IC50 = 2 nM T40016 C6J4SB 57395657 EC50 = 17.3 nM T40016 CINU04 57396254 IC50 = 8 nM T40016 C1O6JU 57396255 IC50 = 2 nM T40016 CSUH91 57396585 IC50 = 41.3 nM T40016 CSRF70 57396586 IC50 = 305 nM T40016 C4BV3D 57396601 IC50 = 5.8 nM T40016 CG9A3H 57396602 IC50 = 4.4 nM T40016 CU4M9T 57396603 IC50 = 1.69 nM T40016 CA49PX 57398362 IC50 = 57.2 nM T40016 CS2MU7 57398378 IC50 = 46.5 nM T40016 CELN93 57398379 IC50 = 37.9 nM T40016 C24YLG 57399054 Ki = 2.4 nM T40016 C0CNX7 57399075 IC50 = 15.9 nM T40016 C54BJR 57399499 IC50 = 142 nM T40016 CVOB64 57399718 IC50 = 6 nM T40016 CT7X2V 57400021 IC50 = 68.7 nM T40016 C4B8RP 57400033 IC50 = 69.3 nM T40016 C0FA2Q 57400034 IC50 = 6 nM T40016 CACH70 57400817 EC50 = 535 nM T40016 CM29BO 57400818 IC50 = 1.9 nM T40016 CY7IE5 57400819 IC50 = 18 nM T40016 CG9KZ2 57400871 EC50 = 14.1 nM T40016 CF83VM 57401459 Ki = 1.94 nM T40016 CJ4LR2 57401460 Ki = 15.7 nM T40016 C7W3YD 57401479 IC50 = 39 nM T40016 C4GIL8 57401833 IC50 = 11.4 nM T40016 C84EUP 57402578 EC50 = 50 nM T40016 CQB6W2 57402579 IC50 = 3.7 nM T40016 C6RX7O 57403004 IC50 = 45 nM T40016 C6IPK0 57403199 Ki = 0.67 nM T40016 CR6L7E 57403222 IC50 = 49 nM T40016 CG2J6D 57403536 IC50 = 7.3 nM T40016 C81TNW 57403537 IC50 = 13.5 nM T40016 C86WRQ 57403538 IC50 = 43.8 nM T40016 CDP21S 57403554 IC50 = 36 nM T40016 C7NX0F 57432086 IC50 = 13.4 nM T40016 CLP69J 57432087 IC50 = 17 nM T40016 CPU6W7 57473898 IC50 = 35 nM T40016 CEJ25K 57473899 IC50 = 10 nM T40016 CUJ08D 57474008 IC50 = 10 nM T40016 C2U1GQ 57524309 IC50 = 125 nM T40016 C3NHX4 57651527 IC50 = 97 nM T40016 CR2J4D 57651532 IC50 = 1600 nM T40016 CW1XC2 57651533 IC50 = 23 nM T40016 C0MTP4 57651538 IC50 = 75 nM T40016 CJ1B4P 57651564 IC50 = 18 nM T40016 CBY05F 57651578 IC50 = 80 nM T40016 C7P3UH 57651588 IC50 = 240 nM T40016 C2QG9T 57651604 IC50 = 42 nM T40016 CJD46O 57651617 IC50 = 410 nM T40016 CSV5U6 57651649 IC50 = 160 nM T40016 CD74EG 57651658 IC50 = 220 nM T40016 COUM81 57666295 Ki = 2.6 nM T40016 CO02KN 57666296 Ki = 4.1 nM T40016 C9Y5ZN 57666298 Ki = 4.6 nM T40016 CQF1I7 57666299 Ki = 1.7 nM T40016 CKS5N7 57666309 Ki = 4.4 nM T40016 C3WG0L 57666312 Ki = 0.5 nM T40016 CB4Y7X 57666322 Ki = 2.4 nM T40016 CS5W9Q 57666329 IC50 = 2.3 nM T40016 CK1PB7 57666331 Ki = 15 nM T40016 C2WL8X 57666350 IC50 = 0.4 nM T40016 CR0F3Y 57666355 IC50 = 0.1 nM T40016 CBDI87 57666363 Ki = 3.1 nM T40016 CBMZ45 57666378 Ki = 2.7 nM T40016 C43GDR 57666397 IC50 = 1.1 nM T40016 CNX5C4 57666415 Ki = 1.9 nM T40016 CZX0O6 57690890 IC50 = 6.9 nM T40016 CN6Q0O 57690891 IC50 = 28 nM T40016 CTM6K5 57690900 IC50 = 7.2 nM T40016 CV0WT1 57690902 IC50 = 3.8 nM T40016 CHDO84 57690904 IC50 = 8.8 nM T40016 C6PKR9 57690906 IC50 = 2 nM T40016 CD5T6X 57690907 IC50 = 4.1 nM T40016 CH45LN 57736637 Ki > 100 nM T40016 C1KZT3 57906156 IC50 > 10000 nM T40016 C3IN9F 57983276 IC50 > 10000 nM T40016 CJ6Y1B 58026134 IC50 = 27 nM T40016 CV1RX3 58026153 IC50 = 28 nM T40016 C19XQV 58026164 IC50 = 2 nM T40016 CR7H3O 58026170 IC50 = 140 nM T40016 C7XL3D 58026176 IC50 = 19 nM T40016 C8S3EQ 58064714 IC50 = 2770 nM T40016 CL42XF 58064726 IC50 = 4800 nM T40016 CPL9A6 58064729 IC50 > 10000 nM T40016 CA0SH5 58064735 IC50 > 10000 nM T40016 C47AUR 58392644 Ki = 0.76 nM T40016 CLU6V4 58392650 Ki = 0.57 nM T40016 CV6G4D 58392653 EC50 = 248 nM T40016 C9CQS0 58392665 Ki = 0.66 nM T40016 CTMC05 58392676 Ki = 0.39 nM T40016 CXF39M 58392685 Ki = 4.8 nM T40016 C9FK1W 58392705 EC50 = 63.9 nM T40016 CSE2H6 58392714 Ki = 0.52 nM T40016 C7FXH3 58392721 Ki = 1.1 nM T40016 C9IAL0 58392730 Ki = 0.71 nM T40016 CBY7Q3 58392757 Ki = 0.57 nM T40016 CWX3L0 58392759 EC50 = 1.3 nM T40016 CJDN90 58392790 Ki = 0.62 nM T40016 CC5L9W 58392802 Ki = 9.8 nM T40016 CO59DQ 58392803 EC50 = 45 nM T40016 CD9V7K 58392806 EC50 = 54.9 nM T40016 C0AZ1T 58392807 Ki = 0.66 nM T40016 CE5S4N 58392813 EC50 = 15.2 nM T40016 C1U8YQ 58392816 Ki = 0.66 nM T40016 CJH51L 58392825 Ki = 1.9 nM T40016 C4C2FT 58599563 IC50 = 7 nM T40016 CWAD17 58731166 Ki <= 500 nM T40016 CI7XQ5 58731245 Ki <= 500 nM T40016 CI6XF5 58742295 IC50 = 0.6 nM T40016 CVGS24 58742335 IC50 = 100 nM T40016 CNW46Q 58742348 IC50 = 211 nM T40016 CUAY18 58742377 IC50 = 22 nM T40016 C4I8UG 58742381 IC50 = 38 nM T40016 CRYK21 58742385 IC50 = 0.79 nM T40016 C0JL7A 58973277 IC50 = 1.15 nM T40016 CV8B1K 59233333 Ki = 69 nM T40016 CN3YR2 59233334 Ki = 35 nM T40016 CY38HG 59233337 Ki = 35 nM T40016 CUX4E7 59233347 Ki = 46 nM T40016 CO63VJ 59233364 Ki = 53 nM T40016 CW3Z2B 59251049 EC50 = 977 nM T40016 C3VD2R 59251055 Ki = 1.51 nM T40016 C14FAP 59251075 Ki = 2 nM T40016 CTZ10A 59251088 Ki = 1.9 nM T40016 C2A9JO 59251119 Ki = 0.81 nM T40016 CHM67D 59251186 Ki = 1.15 nM T40016 C14OUW 59252742 Ki = 7.2 nM T40016 CN4J2B 59252759 Ki = 21 nM T40016 CL91EP 59252761 Ki = 8.1 nM T40016 CZW0C6 59252766 Ki = 36 nM T40016 COH4C0 59252776 Ki = 47 nM T40016 CE9PF6 59252796 Ki = 21 nM T40016 C0WL5E 59252800 Ki = 9.8 nM T40016 CR24NL 59252804 Ki = 19 nM T40016 CR3D9I 59252811 Ki = 46 nM T40016 CV49FS 59252819 Ki = 8.8 nM T40016 C1IOL3 59252821 Ki = 7.5 nM T40016 C5F8SX 59252827 Ki = 1.9 nM T40016 CVT75O 59252830 Ki = 29 nM T40016 C4EV6L 59252842 Ki = 84 nM T40016 CWUE23 59252846 Ki = 7 nM T40016 CA3W0U 59252850 Ki = 1.1 nM T40016 C9F3JN 59252853 Ki = 14 nM T40016 C5B9WH 59252854 Ki = 12 nM T40016 C4K3RM 59252869 Ki = 10 nM T40016 CTM0O8 59252882 Ki = 13 nM T40016 C1VDO0 59266722 IC50 = 1.1 nM T40016 CN6CO4 59272917 IC50 = 0.21 nM T40016 C10MEG 59272918 IC50 = 0.92 nM T40016 CM2L1N 59272923 IC50 = 0.19 nM T40016 CIDC27 59339621 IC50 = 0.04 nM T40016 CQF0V6 59339664 IC50 = 0.02 nM T40016 CF0CQ2 59339738 IC50 = 0.09 nM T40016 CORQ09 59339810 IC50 = 0.029 nM T40016 CC3QG0 59419621 Ki = 18 nM T40016 C4NHO7 59419641 Ki = 5 nM T40016 CYZI85 59556974 IC50 > 10000 nM T40016 C5DU8H 59612841 Ki < 1 nM T40016 CMR3W0 59769897 Ki > 100 nM T40016 C5C3AO 59770003 Ki = 0.226 nM T40016 C9CF2N 59770543 Ki > 100 nM T40016 CI8JB6 59786564 IC50 = 44 nM T40016 C1OE0C 59786572 IC50 = 2.8 nM T40016 COM20D 59786577 IC50 = 100 nM T40016 CH3QT2 59786587 IC50 = 6.6 nM T40016 C2TNO8 60026286 IC50 = 560 nM T40016 CZE5J8 60026377 IC50 = 8 nM T40016 CJ34GW 60026481 IC50 = 59 nM T40016 CJ7E6C 60026483 IC50 = 2 nM T40016 C0LDS2 60026592 IC50 = 11 nM T40016 C31PTC 60026641 IC50 = 9 nM T40016 C67NSE 60026675 IC50 = 13 nM T40016 C6GP5R 60026731 IC50 = 5 nM T40016 C5M8HV 60026772 IC50 = 5 nM T40016 CI36XS 60026787 IC50 = 2 nM T40016 C3JD8M 60026802 IC50 = 14 nM T40016 CE9MI4 60026817 IC50 = 5 nM T40016 C3UQ8M 60026849 IC50 = 7 nM T40016 C04EKW 60026878 IC50 = 18 nM T40016 CM3Y0X 60026895 IC50 = 22 nM T40016 CH5CQ7 60202645 Ki = 4 nM T40016 CIX6M8 66549685 Ki = 19 nM T40016 C5TKZ8 66549686 Ki = 7 nM T40016 C7T5RU 66549878 Ki = 5 nM T40016 C9YN2F 66549879 Ki = 11 nM T40016 C3WQ9J 66549880 Ki = 11 nM T40016 C7DF3G 66549881 Ki = 8 nM T40016 C64VNT 66549882 Ki = 3 nM T40016 C4WER8 66549883 Ki = 557 nM T40016 C69DEI 66550094 Ki = 22 nM T40016 COY2Q0 66550095 Ki = 400 nM T40016 C3THV1 66550096 Ki = 24 nM T40016 C4KM3Y 66550097 Ki = 18 nM T40016 CNDC81 66550098 Ki = 49 nM T40016 CR8X7I 66550099 Ki > 50 nM T40016 CE3QS0 66550320 Ki = 139 nM T40016 C5RMY8 66550321 Ki = 188 nM T40016 CB0VD7 66550322 Ki = 21 nM T40016 CT90BP 66550324 Ki = 8 nM T40016 CSU9T5 66550325 Ki = 28 nM T40016 CJKH71 66550524 Ki = 9 nM T40016 CZ47TU 66550726 Ki = 19 nM T40016 CIN7W5 66550727 Ki = 9 nM T40016 CH7JS8 66550729 Ki = 16 nM T40016 C1CXY9 66996546 IC50 > 10000 nM T40016 CH39DP 67053383 IC50 = 70 nM T40016 C3LF8O 67053425 IC50 = 100 nM T40016 CU5C7T 68327007 Ki > 50 nM T40016 C4UC3D 68833523 IC50 = 0.3 nM T40016 C35MCV 69075970 IC50 = 1800 nM T40016 CNQ8T5 69571559 IC50 = 10 nM T40016 CP7ME8 70681366 IC50 = 5.57 nM T40016 C28NIR 70681401 IC50 = 101 nM T40016 CO2V3L 70681433 IC50 = 29.2 nM T40016 CQ0Z1H 70682700 IC50 = 1642 nM T40016 CEK7F6 70683461 IC50 = 0.63 nM T40016 C5YF1S 70683462 IC50 = 1.5 nM T40016 C0Y7VR 70683502 IC50 = 400 nM T40016 CK8H0A 70683527 IC50 = 0.32 nM T40016 C1V8BT 70683528 IC50 = 0.6 nM T40016 CLCX98 70684785 IC50 = 235 nM T40016 CARO49 70685018 Ki = 0.17 nM T40016 CJIF98 70685568 IC50 = 6.6 nM T40016 CV6S0D 70685569 IC50 = 3.12 nM T40016 C9A4VY 70685580 IC50 = 3.43 nM T40016 CK3U2R 70685600 IC50 = 2.1 nM T40016 C0A5RP 70685628 IC50 = 0.5 nM T40016 CT08DF 70685651 IC50 = 22.1 nM T40016 CJ31YF 70687711 IC50 = 4.4 nM T40016 CZLJ82 70687712 IC50 = 7.3 nM T40016 CCR59B 70687725 IC50 = 7.5 nM T40016 C65IRX 70687751 IC50 = 107 nM T40016 C2DIO4 70687776 IC50 = 1.8 nM T40016 C3K1FC 70687805 IC50 = 4.3 nM T40016 CSZA04 70687806 IC50 = 6.6 nM T40016 C8BEI2 70687807 IC50 = 14.9 nM T40016 C0AEY1 70689007 IC50 > 10000 nM T40016 C6QW5H 70689008 IC50 = 46 nM T40016 C2HP8J 70689009 IC50 = 801 nM T40016 C52VZQ 70689010 IC50 = 1278 nM T40016 C1GCA5 70689011 IC50 = 1601 nM T40016 CD29ZL 70689757 IC50 = 14.8 nM T40016 CA2Z5T 70689778 IC50 = 44.7 nM T40016 CKJ64D 70689802 IC50 = 86.4 nM T40016 C4JUQ2 70689803 IC50 = 88.7 nM T40016 CZ8XA6 70689821 IC50 = 18.3 nM T40016 C2X4VH 70689840 IC50 = 4.7 nM T40016 CH74ZQ 70689841 IC50 = 127 nM T40016 CWR1T7 70691113 IC50 = 1910 nM T40016 CE41BJ 70691114 IC50 = 722 nM T40016 CWK43T 70691115 IC50 = 96 nM T40016 CM1WP7 70691918 IC50 = 28.8 nM T40016 CA2U1S 70691919 IC50 = 3.7 nM T40016 C4NC7P 70691920 IC50 = 2.8 nM T40016 CSRB01 70691940 IC50 = 179 nM T40016 CT45PM 70691941 IC50 = 2.9 nM T40016 C8MHT9 70691942 IC50 = 30.5 nM T40016 CD19KG 70691967 IC50 = 1.99 nM T40016 CPH9W3 70691968 IC50 = 1.6 nM T40016 CT7KY2 70691995 IC50 = 26.7 nM T40016 C7PKB1 70691996 IC50 = 27.2 nM T40016 C32MBT 70693235 IC50 = 820 nM T40016 CXI23M 70693236 IC50 = 4.6 nM T40016 CX0IR5 70693237 IC50 = 1256 nM T40016 CE02OB 70693238 IC50 = 298 nM T40016 CLE0R8 70693239 IC50 = 111 nM T40016 CXA43E 70693965 IC50 = 4.7 nM T40016 CYO30E 70693966 IC50 = 0.89 nM T40016 CE60JR 70693992 IC50 = 1.06 nM T40016 CF4D9M 70694011 IC50 = 1.89 nM T40016 C6ZK1Y 70695317 IC50 = 1423 nM T40016 C9SPT1 70696092 IC50 = 12.4 nM T40016 CI4EG2 70696161 IC50 = 8.9 nM T40016 CE7P8B 70696162 IC50 = 61.3 nM T40016 CBJ0D6 70697330 IC50 > 9000 nM T40016 CGLJ86 70697331 IC50 = 1200 nM T40016 C9QTP1 70697332 IC50 = 4.5 nM T40016 C5QPC0 70697572 Ki = 0.21 nM T40016 CUH71V 71239417 IC50 > 1000 nM T40016 C95CVQ 71245268 Ki = 0.67 nM T40016 C9GC3P 71245282 Ki = 0.52 nM T40016 CM90EO 71245304 Ki = 0.52 nM T40016 CV1QJ5 71245432 Ki = 0.71 nM T40016 C1W0KS 71245462 Ki = 0.57 nM T40016 CP0C6L 71245590 Ki = 0.52 nM T40016 C0NWE2 71451108 Ki = 155 nM T40016 C94FCP 71452686 IC50 = 2300 nM T40016 C8OT4U 71452929 Ki < 1 nM T40016 C0BFS4 71452930 Ki = 58 nM T40016 CLRN15 71452931 Ki > 400 nM T40016 CF7G5Q 71454032 Ki = 98 nM T40016 C35HYI 71456433 Ki = 2 nM T40016 CLM4X2 71456434 Ki = 3 nM T40016 CF08ME 71457470 Ki = 669 nM T40016 C15EYZ 71457556 Ki > 1500 nM T40016 CJR7C5 71460130 Ki = 15 nM T40016 C39VNO 71460131 Ki = 1 nM T40016 CUZQ62 71460135 Ki > 400 nM T40016 CEO5G4 71461616 IC50 = 2800 nM T40016 CHEM26 71461848 Ki = 40 nM T40016 C1MHC0 71467246 IC50 = 6900 nM T40016 C4B0IC 71467248 IC50 = 5800 nM T40016 CVB70W 71508604 EC50 = 2090 nM T40016 CGS13D 71508641 EC50 = 1440 nM T40016 CG6ZR3 71508642 EC50 > 10000 nM T40016 C82UIW 71508688 EC50 = 90 nM T40016 CQCD26 71508715 EC50 = 1500 nM T40016 C13ALQ 71508716 EC50 > 10000 nM T40016 CT52JE 71508749 EC50 > 10000 nM T40016 CV0F5Y 71508789 EC50 = 2810 nM T40016 COI72X 71508790 EC50 = 550 nM T40016 C9XHS2 71508832 EC50 = 690 nM T40016 C92GOZ 71508833 EC50 = 350 nM T40016 CYW34A 71519686 IC50 = 3400 nM T40016 CGK4S8 71543393 Ki > 6020 nM T40016 C83YJF 71544946 IC50 > 5000 nM T40016 CT9Y5D 71549558 IC50 = 3800 nM T40016 C8ZX0F 71549573 IC50 = 11000 nM T40016 CZ8Y7O 71549829 IC50 = 4900 nM T40016 CPFL57 71549843 EC50 > 20000 nM T40016 CY8SP0 71549969 IC50 = 17000 nM T40016 CX6JR5 71550242 IC50 = 3100 nM T40016 C6WIA2 71550244 IC50 = 3000 nM T40016 CSHT69 71550657 IC50 > 5000 nM T40016 C1JP3D 71712294 Ki = 0.7 nM T40016 C0B6GE 71716762 EC50 > 10000 nM T40016 CRDK79 71717362 EC50 = 6200 nM T40016 C5NU0T 71721539 IC50 = 32500 nM T40016 CP5KM8 72163477 IC50 > 10000 nM T40016 CA6O4K 72163478 IC50 > 10000 nM T40016 C27XWS 72163479 IC50 = 4700 nM T40016 C6M9CN 72163480 IC50 = 3800 nM T40016 CL8AH4 72163481 IC50 > 10000 nM T40016 CB2SD9 72163621 IC50 = 2000 nM T40016 CU6NA8 72163622 IC50 = 2100 nM T40016 CTEV75 72163623 IC50 = 1600 nM T40016 CER73F 72163624 IC50 = 2200 nM T40016 CC8VM7 72163625 IC50 > 10000 nM T40016 CS69AC 72163626 IC50 = 9100 nM T40016 CAJ0H5 72163627 IC50 = 4900 nM T40016 C1D3EU 72163754 IC50 = 5000 nM T40016 C1G3ES 72163755 IC50 = 1100 nM T40016 C92WND 72188913 Ki = 13 nM T40016 CP8AC2 72188914 EC50 = 2.4 nM T40016 CA6FO5 72188915 Ki = 6.7 nM T40016 C0IZU8 72188916 EC50 = 0.5 nM T40016 C8UT9I 72188920 Ki = 15 nM T40016 CMKD06 72188921 Ki = 85 nM T40016 C85XAF 72189208 Ki = 7.9 nM T40016 C8ETZ0 72189209 Ki = 4 nM T40016 C1ERA6 72192163 Ki = 0.16 nM T40016 C8IUW4 72192289 Ki = 2.7 nM T40016 CG7D0N 72192290 Ki = 0.9 nM T40016 C34FBN 72544603 IC50 = 2195 nM T40016 CJ62YO 72547740 Ki = 0.12 nM T40016 C4K8DR 72547975 Ki = 0.22 nM T40016 CPA19X 72548209 Ki = 0.83 nM T40016 CN48HM 72548212 Ki = 0.23 nM T40016 C7IA0J 72548214 Ki = 0.14 nM T40016 CJ34IN 72548216 Ki = 0.14 nM T40016 CBF76T 72548443 Ki = 0.16 nM T40016 CELT72 72548445 Ki = 0.17 nM T40016 C8F9MA 72548670 Ki = 0.41 nM T40016 CY9HV3 72548678 Ki = 0.21 nM T40016 CO1PV2 72548922 Ki = 0.13 nM T40016 CV4G5E 72548925 Ki = 0.21 nM T40016 CX7CM5 72549154 Ki = 0.14 nM T40016 CZBE28 72549155 Ki = 0.25 nM T40016 C8JTK6 72549156 Ki = 0.19 nM T40016 CG06BL 72549381 Ki = 28 nM T40016 C1XGF0 72549624 Ki = 0.22 nM T40016 CSC10N 72549625 Ki = 0.73 nM T40016 CN3W7R 72549852 Ki = 10 nM T40016 COFJ20 72549853 Ki = 69 nM T40016 CT0RY5 72550282 Ki = 0.1 nM T40016 CJ48YS 72550284 Ki = 0.21 nM T40016 C6S3FW 72550951 Ki = 0.14 nM T40016 C1C6SR 72551176 Ki = 0.14 nM T40016 CLA3Y9 72710581 Ki = 0.268 nM T40016 CXB45U 72724690 IC50 = 2 nM T40016 CI2K6C 72725442 IC50 = 83 nM T40016 C0W2UD 72725443 IC50 = 23 nM T40016 CQ5D1B 72725444 IC50 = 230 nM T40016 C2PJV7 72725445 IC50 = 110 nM T40016 CQ4Z2C 72725446 IC50 = 10 nM T40016 C47IMQ 72725447 IC50 = 160 nM T40016 CJSK52 72725491 IC50 = 11 nM T40016 CS6J4T 72725492 IC50 = 48 nM T40016 C41FYD 72725493 IC50 = 10 nM T40016 CUG96L 72725494 IC50 = 10 nM T40016 CFHJ16 72725495 IC50 = 78 nM T40016 CW7IY3 72725496 IC50 = 62 nM T40016 CSV1I7 72725497 IC50 = 15 nM T40016 COV09R 72725548 IC50 = 25 nM T40016 CTE01I 72725549 IC50 = 250 nM T40016 C09ZFS 72725550 IC50 = 89 nM T40016 C2Z7QT 72725551 IC50 = 3 nM T40016 C0K2CP 72725552 IC50 = 120 nM T40016 C37MEN 72725553 IC50 = 27 nM T40016 CYSM01 72725554 IC50 = 23 nM T40016 C3POU0 72736045 EC50 = 0.1 nM T40016 CFQK42 73051162 Ki = 0.14 nM T40016 CL3MJ4 73051163 Ki = 0.08 nM T40016 C45NKJ 73051309 Ki = 0.2 nM T40016 CZ2AM8 73051786 Ki = 0.23 nM T40016 CN7CI1 73346216 Ki = 1.42 nM T40016 CPQY04 73346217 Ki = 2.4 nM T40016 CYU73F 73346218 Ki = 285 nM T40016 CW93GP 73346219 Ki = 196 nM T40016 C3A9QB 73346225 Ki = 11 nM T40016 CCJ4V5 73349253 EC50 = 0.66 nM T40016 C0MTX8 73350834 Ki = 2.3 nM T40016 CW0Q8A 73350835 Ki = 3.6 nM T40016 C9LSH7 73350845 Ki = 17 nM T40016 C5YC4W 73352322 Ki = 0.93 nM T40016 CI16HS 73353799 Ki = 17 nM T40016 C2X6KY 73355320 Ki = 0.87 nM T40016 C02PXY 73356866 Ki = 1.3 nM T40016 COU49R 76314656 IC50 = 5 nM T40016 C95NBT 76314657 IC50 = 21 nM T40016 CD7TQ2 76314998 IC50 = 260 nM T40016 CZ08OF 76317198 IC50 = 120 nM T40016 CR5B2V 76317199 IC50 = 15 nM T40016 C5YFZ6 76318225 IC50 = 11 nM T40016 CS25MH 76318649 IC50 = 62 nM T40016 CG3HM7 76321650 Ki > 100 nM T40016 C0RK5D 76321918 IC50 = 13 nM T40016 C7GI5W 76328818 Ki > 100 nM T40016 C3IC5B 76329113 IC50 = 840 nM T40016 C1RB6X 76329114 IC50 = 9 nM T40016 C8NUF6 76329495 IC50 = 270 nM T40016 CP8M1Z 76332766 IC50 = 5 nM T40016 CKDI18 76332767 IC50 = 8 nM T40016 CW35KY 76336757 IC50 = 17 nM T40016 CK21EY 77461202 IC50 = 2 nM T40016 CIU65X 86280440 Ki = 1.22 nM T40016 CZLU45 86710000 Ki = 0.48 nM T40016 CJ6Q7K 86710002 Ki = 4.6 nM T40016 CT50AL 87539277 IC50 = 39.81 nM T40016 CAVY94 87591264 IC50 = 2.1 nM T40016 CY05IC 87733533 IC50 = 3.981 nM T40016 CBH60W 89400603 Ki = 0.52 nM T40016 C9EH7I 89500376 Ki = 2390 nM T40016 C0EQS7 89501406 Ki > 3120 nM T40016 C8JG7O 89510193 Ki = 462 nM T40016 C0VB9S 89953995 Ki = 12 nM T40016 CK29LG 89954151 Ki = 7.6 nM T40016 CFKJ67 89954179 Ki = 0.88 nM T40016 CP68TD 89954189 Ki = 3.1 nM T40016 C6HPE2 89954292 Ki = 31 nM T40016 CPHU03 89954366 Ki = 1.3 nM T40016 C2MPT3 89954418 Ki = 0.64 nM T40016 C0PU6X 89954457 Ki = 0.29 nM T40016 CM38BS 89954484 Ki = 9.7 nM T40016 CQ5WA1 89954525 Ki = 0.15 nM T40016 CU45GK 89954608 Ki = 0.32 nM T40016 CIX49O 89954622 Ki = 11 nM T40016 CXW1Q6 89954759 Ki = 0.59 nM T40016 C90OKR 89954788 Ki = 0.19 nM T40016 CKMB42 89954841 Ki = 0.29 nM T40016 CDH31J 89954858 Ki = 6.6 nM T40016 C9A4ZX 89955032 Ki = 0.42 nM T40016 C4HDM0 89955037 Ki = 0.33 nM T40016 CM5V8H 89955158 Ki = 0.32 nM T40016 CK5D1A 90395281 IC50 > 20000 nM T40016 CQ06RH 90654508 IC50 = 1300 nM T40016 C6VZ7X 90656360 IC50 > 10000 nM T40016 CNCB43 90656361 IC50 > 10000 nM T40016 C4BA8W 90656430 IC50 = 32000 nM T40016 C0Q5MF 90656551 IC50 = 10000 nM T40016 CQM94C 90656552 IC50 = 10000 nM T40016 CA95DL 90656553 IC50 > 10000 nM T40016 C7G4UN 90656554 IC50 > 10000 nM T40016 CXK9Q8 90656555 IC50 > 10000 nM T40016 CJ1X6I 90656556 IC50 = 32 nM T40016 CC0E1Z 90656557 IC50 = 85 nM T40016 CHI35V 90662883 EC50 = 21.1 nM T40016 CA9PL8 91663316 IC50 = 22300 nM T40016 CE4Z3U 102313488 IC50 = 10000 nM T40016 CF67IH 117917065 EC50 = 3.2 nM T40016 CFG2T8 117917077 Ki = 69.4 nM T40016 CDZ31K 117917098 Ki = 1.5 nM T40016 CW27MY 118063735 EC50 > 10000 nM T40016 C6BQ8K 118092322 Ki = 60 nM T40016 C43QTL 118092331 Ki = 120 nM T40016 CZ7DT3 118092342 Ki = 24 nM T40016 CL47CF 118092345 Ki = 44 nM T40016 CGD29J 118092358 Ki = 68 nM T40016 CSK83H 118092376 Ki = 34 nM T40016 CD7RS9 118599615 Ki = 31.62 nM T40016 C70AOV 118599714 Ki = 630.96 nM T40016 C8XLO9 118599727 Ki = 2511.89 nM T40016 CW7G4T 118599742 Ki = 125.89 nM T40016 C9L5EW 118599756 Ki = 5011.87 nM T40016 CVIW94 118599769 Ki = 316.23 nM T40016 CFS28Y 118599779 Ki = 3162.28 nM T40016 CREN83 118707969 Ki = 2.5 nM T40016 CC2I1P 118707970 Ki = 12.9 nM T40016 C7XD9E 118707971 Ki = 8.5 nM T40016 CF60IG 118707972 Ki = 8.7 nM T40016 CZB1G7 118707973 Ki = 110.5 nM T40016 C3XOR9 118707974 Ki = 6.9 nM T40016 CDA17Q 118707975 Ki = 5.7 nM T40016 CTKA86 118707976 Ki = 8.7 nM T40016 CVW2B3 118707977 Ki = 7.4 nM T40016 CLS7C1 118707978 EC50 = 1.2 nM T40016 C9LV0M 118707979 Ki = 1.6 nM T40016 CV4DC0 118707980 Ki = 0.7 nM T40016 COJB29 118707981 Ki = 1.9 nM T40016 C3TLR1 118707982 EC50 = 0.6 nM T40016 CMW3N5 118707983 Ki = 2 nM T40016 C72VHF 118707984 Ki = 7.3 nM T40016 C06ZWX 118707985 Ki = 4 nM T40016 C6Y5JG 118723171 IC50 = 300 nM T40016 CE3I9T 118723172 IC50 = 24 nM T40016 C13AIC 118723173 IC50 = 21 nM T40016 C21SWI 118723174 IC50 = 56 nM T40016 CKR24J 118723175 IC50 = 60 nM T40016 C28YZF 118723176 IC50 = 170 nM T40016 C6AGI7 118723177 IC50 > 2000 nM T40016 C4QO8E 118723178 IC50 = 260 nM T40016 C31RJM 118735258 IC50 = 5.2 nM T40016 C1IC6W 118735259 IC50 = 47 nM T40016 C70CMF 118735260 IC50 = 20.1 nM T40016 C6FDB4 118735261 IC50 = 35.4 nM T40016 C20TNQ 118735262 IC50 = 650 nM T40016 CKWU27 118735263 IC50 = 79 nM T40016 CVZ95N 118735264 IC50 = 28 nM T40016 CLE9O2 121248060 IC50 = 1.7 nM T40016 CPVF94 121248184 EC50 = 5.6 nM T40016 C61QKR 121248207 EC50 = 2.7 nM T40016 CG13LX 122178361 IC50 = 2900 nM T40016 C9LIR4 122179356 Ki = 16 nM T40016 CUI57B 122179357 IC50 < 30 nM T40016 C9U1QL 122179358 Ki = 146 nM T40016 CTQZ35 122179359 Ki = 106 nM T40016 CR98CI 122179360 Ki = 28 nM T40016 C24FBP 122179361 Ki > 384 nM T40016 CGF74Y 122179362 Ki > 384 nM T40016 C10YVG 122179363 Ki > 384 nM T40016 C0OR2H 122186738 Ki = 654 nM T40016 CU0Y8B 122186739 Ki = 39.8 nM T40016 CWF0Q4 122186740 Ki = 115 nM T40016 CBE6Q8 122186741 Ki = 2.67 nM T40016 CX13DR 122186742 Ki = 0.543 nM T40016 CJ74HX 122186743 Ki = 53.7 nM T40016 C05VWL 122186744 Ki = 1.32 nM T40016 CNX5H4 122186745 Ki = 5.45 nM T40016 C4E5JI 122186746 Ki = 1410 nM T40016 CQ6BG8 122186747 Ki = 5.04 nM T40016 CH8O2M 122186748 Ki = 3.06 nM T40016 C4LRN1 122186749 Ki = 94.6 nM T40016 CN9C2T 122192181 IC50 > 31622.78 nM T40016 CCK36V 127029882 IC50 > 5000 nM T40016 CFY1P0 127029884 IC50 = 651 nM T40016 CLDC46 127031152 IC50 > 37000 nM T40016 C60SMC 127031153 IC50 > 12000 nM T40016 CWG34O 127036544 Ki = 0.47 nM T40016 CY0WZ9 129295280 IC50 = 5.6 nM T40016 C65RIZ 129295282 IC50 = 33.6 nM T40016 CM62UE 129295287 IC50 = 14.6 nM T40016 CR23ZG 129295311 IC50 = 47.2 nM T40016 C2LVO7 129295370 IC50 = 57.9 nM T40016 CTI04S 129295372 IC50 = 52.1 nM T40016 C4G2ID 129304679 IC50 = 16.1 nM T40016 CGK48C 129304682 IC50 = 43 nM T40016 CEVZ49 129304683 IC50 = 16.6 nM T40016 CM4LD6 129304687 IC50 = 19.5 nM T40016 C6XAZ5 129304688 IC50 = 17.5 nM T40016 C85QXL 129304691 IC50 = 205 nM T40016 CR3YV9 129304702 IC50 = 16.7 nM T40016 CS2UB8 129304733 IC50 = 28 nM T40016 COU93J 129304741 IC50 = 43 nM T40016 C7K2IE 129304748 IC50 = 9.6 nM T40016 C2GJ8T 129304757 IC50 = 13.3 nM T40016 C7MRB5 129304758 IC50 = 7.5 nM T40016 CN0UA7 129304771 IC50 = 48 nM T40016 CBSJ31 129304830 IC50 = 12.4 nM T40016 C1H0UX 129304861 IC50 = 16 nM T40016 C9ELW1 132275097 IC50 = 2.4 nM T40016 C12UNI 132502971 IC50 = 1430 nM T40016 CK3P0W 132502972 IC50 = 3150 nM T40016 CFT2A4 134132246 EC50 = 47 nM T40016 CP7U8D 134133225 IC50 = 0.62 nM T40016 CNE2Y4 134134891 IC50 = 0.9 nM T40016 COYD80 134135818 IC50 = 1.4 nM T40016 C79OUF 134136440 EC50 = 149 nM T40016 CH9KN0 134136493 EC50 = 1861 nM T40016 C4UX7Z 134137342 EC50 = 0.11 nM T40016 C9TG2N 134137487 IC50 = 0.1585 nM T40016 CED46P 134138613 IC50 = 0.07 nM T40016 C8HY9A 134141623 IC50 = 37 nM T40016 CRJ12I 134141987 IC50 = 558 nM T40016 CNS5V7 134144852 EC50 = 280 nM T40016 CS4P3B 134145141 IC50 = 91 nM T40016 CK10EC 134145786 IC50 = 2400 nM T40016 C0XRT2 134146077 IC50 = 0.09 nM T40016 CVS65Y 134148910 EC50 = 265 nM T40016 CTPU54 134149674 EC50 = 100 nM T40016 C46HMP 134149836 IC50 = 455 nM T40016 CM0TA5 134149846 IC50 = 8.83 nM T40016 CD3E2J 134149965 EC50 = 0.04 nM T40016 CX9T1H 134150995 IC50 = 0.4 nM T40016 C87YMA 134156029 IC50 = 1870 nM T40016 CY7ZM4 134157373 EC50 = 240 nM T40016 CNBM96 134157739 IC50 = 84 nM T40016 CD58OH 134157814 EC50 = 0.05 nM T40016 C30HIQ 134415607 IC50 = 12.2 nM T40016 C3Y2NT 134415609 IC50 = 52.2 nM T40016 CQ53DW 134415610 IC50 = 116 nM T40016 CO32XF 134415624 IC50 = 10.3 nM T40016 CRP1C4 134415742 IC50 = 12.7 nM T40016 C1U9HD 134415745 IC50 = 13.9 nM T40016 CB09XQ 134415864 IC50 = 20.6 nM T40016 CU6Y5D 134415868 IC50 = 35.8 nM T40016 C1GY2T 135156251 EC50 > 10000 nM T40016 CY8U6E 135459005 IC50 > 100000 nM T40016 CBA2F6 135513268 IC50 > 50000 nM T40016 CTF0J3 135567449 Ki = 50.12 nM T40016 CN24YZ 135567451 Ki = 251.19 nM T40016 CPF3B4 135567452 Ki = 7.943 nM T40016 C34JMK 135571931 IC50 > 100000 nM T40016 C5MXO2 136000568 Ki = 0.6 nM T40016 CD07ZO 136000655 Ki = 7 nM T40016 CM6OX5 136000656 Ki = 0.8 nM T40016 CZ2D6U 136059148 Ki = 2.2 nM T40016 C6HOU3 136059149 Ki = 2 nM T40016 CE1G9O 136059150 Ki = 3.8 nM T40016 C7LSN6 136088946 EC50 = 0.6 nM T40016 C1F4BY 136088947 Ki = 0.7 nM T40016 CRJ9V5 136088948 IC50 = 3.5 nM T40016 C1M3WU 136088949 Ki = 1.5 nM T40016 CR4X3Q 136088950 Ki = 5.8 nM T40016 CI4RW5 136088951 Ki = 31 nM T40016 C4OX9M 136088952 Ki = 0.4 nM T40016 C2JV0P 136088953 Ki = 2700 nM T40016 C98CLF 136098616 Ki = 5.7 nM T40016 CEP7N9 136254190 IC50 = 3 nM T40016 C1B2KD 137631905 IC50 = 0.156 nM T40016 C38MWL 137632612 IC50 > 1000 nM T40016 CC10WR 137632878 IC50 > 30000 nM T40016 CE48UI 137633773 IC50 > 30000 nM T40016 COI80Z 137634236 IC50 = 12.59 nM T40016 CQ6J5I 137637753 IC50 > 30000 nM T40016 C5B4PZ 137637922 IC50 > 30000 nM T40016 CAHT60 137638938 IC50 > 30000 nM T40016 CPD87Y 137639726 IC50 = 19.95 nM T40016 CGCA32 137639839 IC50 > 30000 nM T40016 CEGX68 137640275 IC50 = 0.12 nM T40016 C8TBZ4 137641110 IC50 = 24.3 nM T40016 CZRS94 137641411 IC50 > 30000 nM T40016 CXQ8P3 137641761 IC50 > 30000 nM T40016 C6E0AL 137642668 IC50 = 5770 nM T40016 C0T3HQ 137643401 IC50 > 30000 nM T40016 C46QZA 137647155 IC50 = 7870 nM T40016 C0K4BJ 137648403 IC50 = 464 nM T40016 C30ZJF 137648477 IC50 = 6.31 nM T40016 CJE8B2 137648715 IC50 > 30000 nM T40016 C4SJD8 137650072 IC50 = 7480 nM T40016 CAS7B9 137651118 IC50 = 3590 nM T40016 CRYF53 137651691 IC50 = 1970 nM T40016 CW9Y6S 137651919 IC50 = 12.7 nM T40016 CWZ06G 137652587 IC50 = 5420 nM T40016 CO92KL 137654415 IC50 = 15.85 nM T40016 C5MXU1 137655191 IC50 = 0.066 nM T40016 C1CM0L 137656584 IC50 > 30000 nM T40016 C75CDY 137658459 IC50 = 2040 nM T40016 CP46JS 137658546 IC50 > 30000 nM T40016 COT7M8 137659850 IC50 > 30000 nM T40016 C7JKI9 137660091 IC50 > 1000 nM T40016 CZ49NM 137660168 IC50 = 2020 nM T40016 CQWG60 137661608 IC50 = 0.15 nM T40016 CZWT36 137661763 IC50 > 30000 nM T40016 C54OHS 137661940 IC50 = 2110 nM T40016 C7EKA2 138911324 IC50 = 8.5 nM T40016 C96ONI 141538600 IC50 = 58.3 nM T40016 CR6Y2I 141538601 IC50 = 28.5 nM T40016 CR5Y9P 145949269 IC50 = 1.93 nM T40016 CW3Y0H 145949340 IC50 > 20000 nM T40016 CP5U7Q 145949975 EC50 = 57 nM T40016 COKU96 145950643 IC50 = 32 nM T40016 CPK5U1 145951022 IC50 > 20000 nM T40016 CKT24R 145951943 IC50 > 20000 nM T40016 CD49VI 145953389 IC50 = 18.1 nM T40016 CU19EN 145958055 IC50 = 11.2 nM T40016 C5U3JV 145958117 IC50 = 8.5 nM T40016 CORP09 145958365 EC50 = 17.4 nM T40016 CR6T8S 145959457 IC50 = 64 nM T40016 CU84AB 145963803 IC50 < 3.2 nM T40016 C9AH5J 145964455 IC50 < 4 nM T40016 C72QDJ 145964714 IC50 = 9.3 nM T40016 CSJ60M 145964914 EC50 = 3.5 nM T40016 C2QB3L 145964915 IC50 < 4.1 nM T40016 CX94YN 145965573 IC50 < 0.34 nM T40016 CF0PO7 145965716 IC50 = 57 nM T40016 CS8G3K 145965784 EC50 = 29 nM T40016 C9Y6RT 145965869 IC50 = 7.1 nM T40016 CE9PD6 145966463 IC50 = 160 nM T40016 CW61TA 145966634 IC50 = 1.6 nM T40016 C14OAC 145966706 IC50 = 2 nM T40016 CVT2B5 145971542 IC50 = 7.2 nM T40016 C1V7EP 145972549 EC50 = 13 nM T40016 C34ENO 145972998 IC50 < 1.6 nM T40016 C71PDT 145973741 IC50 = 21 nM T40016 C8DFZ5 145973994 IC50 = 6.1 nM T40016 C0V1TU 145974260 EC50 = 3.5 nM T40016 CM9QN8 145974940 IC50 = 42 nM T40016 CJFS50 145975057 IC50 = 4.7 nM T40016 C19HXS 145975460 IC50 = 11 nM T40016 C2GUH7 145975580 EC50 = 23 nM T40016 CH87UD 145976543 IC50 = 120 nM T40016 C7CUS0 145976724 IC50 < 0.42 nM T40016 CBOW92 145977353 IC50 = 39 nM T40016 C32VLX 145977741 IC50 = 449 nM T40016 C1PMA8 145977753 EC50 = 87 nM T40016 CJY2W5 145978475 IC50 < 6.8 nM T40016 C5T7IK 147930449 Ki = 316.23 nM T40016 C30SYM 155459658 IC50 = 62 nM T40016 CGB78J 155459666 IC50 = 73.7 nM T40016 C0MF5X 155512827 IC50 = 9.5 nM T40016 C28RHM 155514304 Ki = 1995.26 nM T40016 CE2YJ9 155514399 Ki = 79.43 nM T40016 CQF09V 155516050 Ki = 630.96 nM T40016 CELU49 155517819 Ki > 15848.93 nM T40016 C2E4XV 155518137 Ki = 12589.25 nM T40016 C4QAB0 155518139 Ki > 15848.93 nM T40016 C6VIG2 155518655 IC50 = 1012 nM T40016 CCO0Z4 155519877 Ki = 199.53 nM T40016 CC5JZ4 155520100 IC50 > 1000 nM T40016 COF3R4 155520306 IC50 = 0.41 nM T40016 C8BD6Y 155522508 Ki = 398.11 nM T40016 C71VIK 155525344 Ki = 1258.93 nM T40016 C1WAQ6 155527406 Ki = 1258.93 nM T40016 C5T2QN 155528866 Ki = 158.49 nM T40016 CQM89D 155529443 Ki = 1.585 nM T40016 CR0N3F 155529454 Ki = 125.89 nM T40016 CB0XS4 155529625 Ki > 15848.93 nM T40016 C5Y4FK 155531943 IC50 = 6 nM T40016 C3HFZ6 155534085 Ki > 15848.93 nM T40016 CF52DM 155535034 Ki = 1.259 nM T40016 CXR2W1 155536089 IC50 = 4016 nM T40016 C3FON4 155537084 Ki > 12589.25 nM T40016 CJH5I3 155538097 IC50 = 135 nM T40016 COP7X8 155539171 IC50 > 10000 nM T40016 C78ISM 155540009 IC50 = 202 nM T40016 C28KPU 155540268 IC50 = 20 nM T40016 C84LKI 155540713 IC50 = 130 nM T40016 CIAW80 155544156 IC50 = 1051 nM T40016 C76OVS 155544396 Ki > 12589.25 nM T40016 C25HEV 155545046 IC50 > 1000 nM T40016 CR6UY8 155545121 IC50 = 1644 nM T40016 C1XGF5 155546726 IC50 = 17.6 nM T40016 CC36TR 155546752 IC50 = 89 nM T40016 CJ9T5D 155548288 IC50 = 10 nM T40016 C6H2ML 155552723 Ki = 316.23 nM T40016 CW8BH4 155554673 Ki = 1258.93 nM T40016 C9WV3L 155556878 Ki = 1000 nM T40016 CR5ZI2 155557239 Ki = 1258.93 nM T40016 CPY83L 155558503 Ki > 15848.93 nM T40016 C0FEP8 155559859 IC50 > 1000 nM T40016 CQ7HG2 155561626 Ki = 2.512 nM T40016 CBM45A 155563942 IC50 > 1000 nM T40016 CD4K6Z 155564467 Ki = 19.95 nM T40016 CS25QB 155564604 IC50 = 111 nM T40016 C7YK6N 155565026 IC50 = 870 nM T40016 CPX2J5 155566857 Ki > 15848.93 nM T40016 C79WFJ 155567245 Ki > 15848.93 nM T40016 CME1B7 155567676 Ki = 6309.57 nM T40016 CWQI82 136130172 Ki = 370 nM T40016 D00DNY 3213 IC50 = 90000 nM T40016 D00ZGW 46883841 IC50 = 199.53 nM T40016 D01ETZ 261000 Ki = 9.65 nM T40016 D01NVD 46830196 IC50 = 100 nM T40016 D02UID 16734800 IC50 = 1000 nM T40016 D05XVM 18189209 IC50 = 1937 nM T40016 D05ZUX 44207909 Ki >= 1000 nM T40016 D07KWO 9823099 IC50 = 2.4 nM T40016 D08KQM 24816375 Ki = 2.4 nM T40016 D09FQL 16756780 IC50 = 900 nM T40016 D09OKK 9951771 Ki = 564 nM T40016 D0D6GI 46888441 EC50 = 93 nM T40016 D0EG5G 46888467 EC50 = 19 nM T40016 D0F1SS 44605900 IC50 > 1000 nM T40016 D0GR5L 9906282 Ki = 1.4 nM T40016 D0J7XZ 9819614 Ki = 0.17 nM T40016 D0L5IC 9820558 Ki = 0.1 nM T40016 D0M0RS 11560224 Ki > 1000 nM T40016 D0N8UD 46888391 IC50 = 86 nM T40016 D0O5ZG 44305900 IC50 = 1914 nM T40016 D0PR2T 16756782 IC50 = 13000 nM T40016 D0S9KH 63052 IC50 = 600 nM T40016 D0T2RY 9948320 Ki >= 1000 nM T40016 D0T4SL 72512 IC50 = 90000 nM T40016 D0V4RZ 25113722 IC50 = 7200 nM T40016 D0XS0R 44433505 Ki = 1758 nM T99834 C9SYZ3 3708153 EC50 = 22300 nM T99834 C8PDE1 14686324 EC50 = 42500 nM T99834 C45BQH 132585194 EC50 = 4800 nM T42048 D02YNI 9936746 Ki = 4 nM T42048 D05ICT 132010322 Ki = 4.9 nM T42048 D07OFM 46943432 Ki = 30.3 nM T42048 D0M2TS 71600087 Ki = 12.2 nM T42048 D0PH9I 118693659 Ki = 63.1 nM T42048 D0ZW4W 46907787 Ki = 6.6 nM T42048 D09SFV 3973 IC50 = 13700 nM T42048 C92EYR 1503595 IC50 = 30000 nM T42048 CIG94A 13953713 IC50 = 12589.25 nM T42048 C3VRO9 44557921 IC50 > 10000 nM T42048 C98BLM 49871817 IC50 = 19.1 nM T42048 CG3PR6 52912222 IC50 = 0.631 nM T42048 CBXV52 52932793 IC50 = 316.23 nM T42048 CJE59U 52932930 IC50 = 1258.93 nM T42048 CSZ2T6 52932933 IC50 = 3162.28 nM T42048 CN87IR 52933159 IC50 = 1258.93 nM T42048 CG6OL4 52933160 IC50 = 794.33 nM T42048 CP8Y9K 52933161 IC50 = 1000 nM T42048 CK8Z4P 52933165 IC50 = 3162.28 nM T42048 CKC17F 52933403 IC50 = 1000 nM T42048 CD08ZX 52933405 IC50 = 1000 nM T42048 C1T7VQ 52933407 IC50 = 1258.93 nM T42048 CO8VX9 52933655 IC50 = 1584.89 nM T42048 C6G7BE 52933893 IC50 = 1000 nM T42048 C7VN1E 52934039 IC50 = 501.19 nM T42048 CUZE18 52934122 IC50 = 1000 nM T42048 CN16FE 52934128 IC50 = 1995.26 nM T42048 CTS13B 52934275 IC50 = 630.96 nM T42048 CNOH36 52935183 IC50 = 199.53 nM T42048 CLRH53 52935478 IC50 = 794.33 nM T42048 CJIB35 53054190 IC50 = 4700 nM T42048 C6V8YR 53054191 IC50 = 13000 nM T42048 C09HTR 53054200 IC50 = 1000 nM T42048 CUS8F7 53054236 IC50 = 4800 nM T42048 CX5QN4 53054237 IC50 = 14000 nM T42048 CD2TY9 53054238 IC50 = 6500 nM T42048 C47GAW 53054240 IC50 = 5400 nM T42048 CVH2G1 53054241 IC50 = 2200 nM T42048 CF9E2V 53054248 IC50 = 1900 nM T42048 CRWK92 53054249 IC50 = 5900 nM T42048 CSXI51 53054250 IC50 = 1800 nM T42048 CM12EL 53054251 IC50 = 1900 nM T42048 CY5L3J 53054252 IC50 = 4000 nM T42048 CWV76Y 53054258 IC50 = 700 nM T42048 CIU8P7 53054259 IC50 = 500 nM T42048 CVX3R0 53054274 IC50 = 3000 nM T42048 CB05OM 53054276 IC50 = 1100 nM T42048 CLR97U 53054289 IC50 = 1000 nM T42048 CJ6E2Q 53054291 IC50 = 3300 nM T42048 C1WSZ4 53054297 IC50 = 1500 nM T42048 C7A2XC 53054319 IC50 = 2000 nM T42048 C0J1EO 53054320 IC50 = 3800 nM T42048 CK68UF 53054321 IC50 = 800 nM T42048 CJY5S2 53054322 IC50 = 3200 nM T42048 C1YW5L 53054324 IC50 = 2100 nM T42048 C8Q6WG 53054325 IC50 = 1000 nM T42048 C9V5LX 53318989 IC50 = 220 nM T42048 C1KWY4 54759170 IC50 = 2500 nM T42048 C7HK2C 56924692 IC50 = 1100 nM T42048 CX6SD9 56950289 IC50 = 3000 nM T42048 CZ6NE0 56950420 IC50 = 1400 nM T42048 CJ5BE9 56950421 IC50 = 2200 nM T42048 CL96VQ 56950422 IC50 = 1300 nM T42048 CCLD98 56950423 IC50 = 8600 nM T42048 CZD7G2 56950424 IC50 = 4200 nM T42048 CPQ0B7 56950425 IC50 = 8600 nM T42048 CL90DK 56950426 IC50 = 700 nM T42048 CF9IJ1 56950561 IC50 = 700 nM T42048 CH24QC 56950562 IC50 = 8200 nM T42048 CU62NO 56950563 IC50 = 11000 nM T42048 CRD86M 56950564 IC50 = 11000 nM T42048 CNQ2L5 56950565 IC50 = 21000 nM T42048 CB3A1Z 56950566 IC50 = 8400 nM T42048 C5ADP4 56950567 IC50 = 13000 nM T42048 CFW0D1 57339435 IC50 = 501.19 nM T42048 CF8B4E 60498769 IC50 = 62000 nM T42048 CPY59D 67195867 IC50 = 25118.86 nM T42048 CN3KZ8 68161075 IC50 = 316.23 nM T42048 C49IOA 68161669 IC50 = 398.11 nM T42048 CJ7N3M 68184870 IC50 = 1000 nM T42048 CT4Z2A 68184871 IC50 = 398.11 nM T42048 CEX74I 68186034 IC50 = 5011.87 nM T42048 C25INY 68204735 IC50 = 630.96 nM T42048 CMC7V5 70664240 IC50 = 630.96 nM T42048 C1I6OH 70681167 IC50 = 3162.28 nM T42048 C7GJW9 70681170 IC50 = 316.23 nM T42048 C8H4JX 70681173 IC50 = 501.19 nM T42048 C6NYK2 70681174 IC50 = 398.11 nM T42048 C8KBJ0 70683271 IC50 = 501.19 nM T42048 CXD3F9 70691699 IC50 = 251.19 nM T42048 CL8Y9N 71450297 IC50 = 630.96 nM T42048 C6CQT5 71462842 IC50 = 1584.89 nM T42048 CIPN50 71760902 Ki = 35 nM T42048 C2AFW1 72702849 IC50 = 501.19 nM T42048 C3R1IL 72703043 IC50 = 100000 nM T42048 CK9O6W 72705811 IC50 = 6309.57 nM T42048 C5TB9S 77843982 Ki = 110 nM T42048 CS6XE0 77846025 Ki = 3.2 nM T42048 COZ8S1 78319129 Ki = 290 nM T42048 C4IF8T 78425807 Ki = 10 nM T42048 CFE7R3 86270928 Ki = 10 nM T42048 C53QEW 86669224 IC50 = 6309.57 nM T42048 CEDL57 89657555 IC50 = 7 nM T42048 CZJ8W9 90387575 Ki = 4.2 nM T42048 C1W3XP 112499930 IC50 = 1800 nM T42048 C6A1RW 118120978 IC50 = 1710 nM T42048 CHB87O 118120979 IC50 = 1320 nM T42048 CPN74M 118719856 IC50 = 501.19 nM T42048 CE8DL3 118719857 IC50 = 794.33 nM T42048 COEU47 118719858 IC50 = 1258.93 nM T42048 CX05SW 118719859 IC50 = 630.96 nM T42048 CRCG07 118719860 IC50 = 501.19 nM T42048 C03XDG 118719861 IC50 = 630.96 nM T42048 C3ML2F 118719862 IC50 = 398.11 nM T42048 CZ67WF 118719863 IC50 = 25118.86 nM T42048 C0HR9Y 118719864 IC50 = 501.19 nM T42048 C7F4EP 118719865 IC50 = 316.23 nM T42048 CA40QV 118719866 IC50 = 501.19 nM T42048 CZ8QI6 118719867 IC50 = 1000 nM T42048 C8NRI9 118719868 IC50 = 794.33 nM T42048 C3Y2WT 118719869 IC50 = 794.33 nM T42048 C52HPM 118719870 IC50 = 501.19 nM T42048 CUT97H 118719871 IC50 = 501.19 nM T42048 CBE68N 118719872 IC50 = 1258.93 nM T42048 C29WRE 118719873 IC50 = 501.19 nM T42048 C8J0TY 118719874 IC50 = 1000 nM T42048 CZR10C 118719875 IC50 = 2511.89 nM T42048 C35AWU 118719876 IC50 = 1584.89 nM T42048 C3QJ5L 122181550 IC50 > 50118.72 nM T42048 CO25IW 122191031 IC50 >= 10000 nM T42048 C4WGV6 122191040 IC50 = 10000 nM T42048 CDY43J 122191048 IC50 >= 10000 nM T42048 C4GYP3 126521168 IC50 = 25 nM T42048 CL2PG5 126521180 IC50 = 18 nM T42048 CQV90I 126521354 IC50 = 16 nM T42048 C1DOG4 126521586 IC50 = 10 nM T42048 CRY0S6 126563516 IC50 = 14 nM T42048 CN0D6M 126563562 IC50 = 13 nM T42048 CKB36S 126563576 IC50 = 11 nM T42048 CX79NH 126563597 IC50 = 39 nM T42048 C2K5XG 126563611 IC50 = 23 nM T42048 CZ06NR 126563612 IC50 = 44 nM T42048 CM5P2Z 126563615 IC50 = 36 nM T42048 C15ILF 126564427 IC50 = 10 nM T42048 CHO12Y 126564469 IC50 > 10000 nM T42048 CB2AS4 126564470 IC50 = 9 nM T42048 CBW08I 126564471 IC50 = 19 nM T42048 CD78GB 126564481 IC50 = 21 nM T42048 CNP2L7 126564832 IC50 = 14 nM T42048 C58PNK 126564833 IC50 = 21 nM T42048 CHPV09 126564847 IC50 = 12 nM T42048 CJZW04 126564858 IC50 = 13 nM T42048 CH14FC 127032939 IC50 = 4800 nM T42048 CS4NG8 127033568 IC50 = 31700 nM T42048 C9L1OG 130345579 Ki = 2.5 nM T42048 CRNY32 135397673 Ki = 0.18 nM T42048 CV4X7R 135566898 Ki = 1640 nM T42048 CU2F1G 135566900 Ki = 220 nM T42048 C5F3LV 135567026 IC50 > 100000 nM T42048 CW94QO 136226511 Ki = 240 nM T42048 CO71RI 137285009 IC50 = 2241 nM T42048 CS9MR6 137285011 IC50 = 2193 nM T42048 CFXE14 137321203 IC50 = 31.62 nM T42048 CXN4U1 137321204 IC50 = 1258.93 nM T42048 C4VNB8 137369426 IC50 = 52 nM T42048 CU5N8O 137701509 IC50 = 11200 nM T42048 CQ6XB7 139030526 IC50 = 31622.78 nM T42048 C1G9LA 139035062 Ki = 5.3 nM T42048 CG6X3A 142535938 IC50 = 42 nM T42048 CD6U7X 145925666 IC50 = 246.3 nM T42048 C1HLK5 145951928 IC50 = 21 nM T42048 CV83ED 145972103 Ki = 17 nM T42048 CK20BY 145988169 Ki = 42.4 nM T42048 C9FIY4 153534005 IC50 > 20000 nM T42048 CFD6H1 155352361 IC50 = 51000 nM T42048 CFK2B1 155352401 IC50 = 200000 nM T42048 C76QMK 155513141 Ki = 8.2 nM T42048 C27LFN 155514936 IC50 = 770 nM T42048 C6OP0S 155535292 Ki = 11.1 nM T42048 C0HI7N 155536879 IC50 = 456 nM T42048 CUX25H 155547195 Ki = 13.9 nM T42048 CZA5N1 155561689 IC50 > 20500 nM T42048 C7ICA9 155564455 IC50 = 78 nM T42048 D00XRH 91820725 IC50 = 19952.62 nM T42048 D03LIP 13953710 IC50 = 28.4 nM T42048 D09HBR 135566899 Ki = 100 nM T42048 D09VHS 3971 IC50 = 11500 nM T42048 D0F5TZ 91827383 IC50 = 7943.28 nM T42048 D0N5BI 91668541 IC50 > 50118.72 nM T42048 D0WU1S 52912189 Ki = 7.2 nM T09572 D0A3CL 49801838 IC50 = 27 nM T09572 D0TV4N 9865843 Ki = 5.5 nM T09572 D0U0YR 11520239 IC50 = 3 nM T09572 D00RUE 60169095 IC50 = 20 nM T09572 D03KWP 71660914 IC50 = 48 nM T09572 D0C5RD 71719525 IC50 = 50 nM T09572 D0HH1O 71731806 IC50 = 17 nM T09572 D0MT7T 71816518 IC50 = 6.8 nM T09572 D0Q1NA 71660917 IC50 = 77 nM T09572 D0V8FC 60169096 IC50 = 30 nM T09572 C97FYX 702501 IC50 = 43000 nM T09572 C12OHT 1252415 Ki = 11300 nM T09572 CQ6BS4 2276336 Ki = 8100 nM T09572 CUM8T0 2729098 IC50 = 109 nM T09572 CRA9T2 2729502 Ki = 347 nM T09572 CVE13J 2881764 Ki = 11900 nM T09572 CSM9V8 3410248 IC50 = 114 nM T09572 CX6CF2 3611477 IC50 = 82 nM T09572 C2EN7Y 4219492 IC50 = 59 nM T09572 CB9WS0 4653788 IC50 > 2000 nM T09572 C5I9SA 4826270 Ki = 7800 nM T09572 C39UDN 5312114 IC50 = 3500 nM T09572 CBJD49 5817261 IC50 = 56 nM T09572 CRV52B 6621104 IC50 = 30 nM T09572 CP5X6Z 9799244 EC50 = 96 nM T09572 C5GL6S 9799726 Ki = 29 nM T09572 CA4Z7C 9801165 Ki < 1 nM T09572 C8XGV3 9804849 IC50 = 16 nM T09572 CYIT28 9806086 IC50 = 50 nM T09572 C1NQC6 9807658 IC50 = 4.9 nM T09572 C2MIW9 9821717 IC50 = 2 nM T09572 C5RIY7 9824428 IC50 = 250 nM T09572 C1J9MV 9824856 IC50 = 6 nM T09572 CG3X9R 9828622 IC50 = 300 nM T09572 CJZ9L7 9829942 IC50 = 5 nM T09572 CX2PO5 9844702 IC50 = 17 nM T09572 C0Q8UT 9848699 Ki = 24 nM T09572 C2PU9N 9851676 Ki = 11 nM T09572 CAKP95 9866552 IC50 = 10 nM T09572 CSTG23 9866745 IC50 = 2 nM T09572 C74RZP 9887476 IC50 = 2.7 nM T09572 C34NSZ 9887864 IC50 = 7 nM T09572 C6EK5P 9888078 IC50 > 100 nM T09572 C9BRE3 9895005 Ki = 6.4 nM T09572 CY1P7H 9895868 IC50 = 140 nM T09572 CTZ48N 9910346 IC50 = 1.9 nM T09572 C5YM8X 9915039 Ki = 0.17 nM T09572 CIP6V7 9932896 IC50 = 0.54 nM T09572 C4L1GA 9934033 IC50 = 3.4 nM T09572 CDY39E 9934161 IC50 = 9 nM T09572 CSWJ86 9954518 Ki = 19.95 nM T09572 CTUO16 9955811 IC50 = 1300 nM T09572 CT7AP4 9978378 IC50 = 11 nM T09572 C5FB3N 9978428 IC50 = 5 nM T09572 CMY73F 9978490 IC50 = 7 nM T09572 C9XH3V 9978508 IC50 = 5.5 nM T09572 CF41ZD 9980157 IC50 = 16 nM T09572 C7TPF5 9983233 IC50 = 2 nM T09572 CVL8X0 9984325 Ki = 45 nM T09572 C9Y6GX 9985634 Ki = 9.772 nM T09572 CS6Q2J 9985881 Ki = 34 nM T09572 CV2D9B 9986014 Ki = 14 nM T09572 C4T2XD 9986044 Ki = 10 nM T09572 CP8WR3 9999058 IC50 = 62 nM T09572 CG14IV 10000146 IC50 = 0.9 nM T09572 CQL12P 10004545 Ki = 0.6 nM T09572 C6OI1A 10005009 IC50 = 1.9 nM T09572 C6Q0IN 10007632 Ki = 823 nM T09572 CXL43G 10008279 Ki = 16 nM T09572 CZ45JK 10024145 IC50 = 6 nM T09572 C4U8JG 10024171 IC50 = 5.9 nM T09572 C3O2EL 10024175 IC50 = 15 nM T09572 C8M2YA 10025637 IC50 = 10 nM T09572 C3NPS8 10025899 IC50 = 12 nM T09572 CS14OM 10027853 IC50 = 1.5 nM T09572 CP9JI2 10029161 Ki = 59 nM T09572 C9XTE6 10029835 Ki = 35 nM T09572 CRJ41C 10029836 Ki = 63 nM T09572 C4XK0H 10031575 Ki = 7 nM T09572 C0UQ4M 10036257 IC50 > 2000 nM T09572 CD4KM9 10041636 IC50 = 120 nM T09572 C02OIU 10047339 IC50 = 28 nM T09572 CA2ZW7 10050565 IC50 = 4.1 nM T09572 C4IS6W 10053890 Ki = 25 nM T09572 CGHX74 10053937 Ki = 10.96 nM T09572 CFA8Y5 10054046 Ki = 2600 nM T09572 C5T6CZ 10059666 IC50 > 2000 nM T09572 C0Y9JS 10067783 IC50 = 0.9 nM T09572 C8PH7Y 10070016 IC50 = 11 nM T09572 CM5S6R 10070680 IC50 = 21 nM T09572 C2Z4FO 10073563 IC50 = 790 nM T09572 CCN5S8 10073934 IC50 = 2.9 nM T09572 CRQL64 10075375 IC50 = 4 nM T09572 C3T7HL 10077022 Ki = 1800 nM T09572 CWD1K0 10077403 Ki = 6.8 nM T09572 C1UCY7 10098577 Ki = 38 nM T09572 CR3MJ4 10099409 Ki = 24 nM T09572 C3FME5 10100662 Ki = 16 nM T09572 C2D6TX 10113523 Ki = 1.2 nM T09572 CNCP64 10114686 IC50 = 0.88 nM T09572 CQ3U9H 10115919 Ki = 2.6 nM T09572 C8MJ1U 10117415 Ki = 1.4 nM T09572 CXJ79U 10118862 Ki = 0.31 nM T09572 CT5GK7 10118863 Ki = 0.45 nM T09572 CX4IA7 10126754 EC50 = 380 nM T09572 C7IFU2 10127348 EC50 = 96 nM T09572 CG7Z9I 10128764 Ki = 1428 nM T09572 COS3D1 10128900 Ki = 2.2 nM T09572 CEO59I 10129026 Ki = 281 nM T09572 CW5O4B 10129036 Ki = 52 nM T09572 C3FS7G 10129058 Ki = 18 nM T09572 CJ05QL 10129135 Ki = 76 nM T09572 C1XK6M 10139496 Ki = 15.85 nM T09572 CTND76 10139873 Ki = 100 nM T09572 CDN19U 10140070 Ki = 6 nM T09572 C8MTR3 10140707 Ki = 4.3 nM T09572 CCSW12 10141528 Ki = 5.5 nM T09572 CP9Q6O 10142124 Ki = 2.6 nM T09572 CFL14Q 10142464 Ki = 37 nM T09572 CX9EI2 10143421 Ki = 19 nM T09572 CZ95DQ 10143980 Ki = 15 nM T09572 CPR42N 10149893 IC50 = 8300 nM T09572 CZT7L9 10150552 EC50 = 110 nM T09572 C2L3HU 10150954 EC50 = 210 nM T09572 CD9V8P 10150955 IC50 = 3 nM T09572 C2X9YI 10152629 Ki = 99 nM T09572 C9VP5L 10152726 Ki = 523 nM T09572 CVGB64 10152879 Ki = 4 nM T09572 C9TQ1J 10159452 IC50 = 2.7 nM T09572 CLW3P2 10159789 Ki = 7.4 nM T09572 C2V1TA 10159797 Ki = 19.95 nM T09572 CRW17C 10160079 Ki = 398.11 nM T09572 CBV5S9 10161039 Ki = 1.5 nM T09572 C8ALH2 10164110 Ki = 2.6 nM T09572 CJ5HL7 10165163 Ki = 2.1 nM T09572 CX36LA 10165503 Ki = 2.5 nM T09572 CZQ69G 10165656 Ki = 27 nM T09572 CFQM97 10166038 Ki < 100 nM T09572 C9EJT4 10166088 Ki = 131 nM T09572 C6ZPK7 10173726 IC50 = 4.5 nM T09572 CC2F7Z 10173787 IC50 = 18 nM T09572 CM9KF2 10174522 Ki = 241 nM T09572 CO2XG1 10174940 Ki = 1.6 nM T09572 CH25WF 10174984 Ki = 2 nM T09572 CX48ZP 10184368 Ki = 4.7 nM T09572 CF8Q2N 10185187 Ki = 50 nM T09572 C47RGT 10186370 Ki = 35 nM T09572 CUO81F 10186375 Ki = 5.4 nM T09572 CQP58G 10186594 Ki = 0.98 nM T09572 C80YEW 10188732 Ki = 82 nM T09572 CM0RA3 10195637 Ki = 4.1 nM T09572 CGJ7D9 10195667 Ki = 18 nM T09572 C9OB3S 10196098 Ki = 3 nM T09572 C2K1LR 10196214 Ki = 178 nM T09572 CBX4C2 10196316 Ki = 21 nM T09572 CD9N3H 10196460 Ki = 3 nM T09572 CYT8S5 10196576 Ki = 9 nM T09572 C5EGZ8 10196608 Ki = 16 nM T09572 C0OB2A 10196742 Ki = 49 nM T09572 CV9H1P 10202381 IC50 = 1000 nM T09572 C6M4SO 10203421 Ki = 3.3 nM T09572 C1V9WG 10204047 Ki = 1.1 nM T09572 CUL57F 10204151 Ki = 0.84 nM T09572 C48NGR 10206922 Ki = 5.6 nM T09572 C63SDN 10209344 Ki = 0.63 nM T09572 CMY61O 10210351 Ki = 20 nM T09572 CDK26C 10217978 Ki = 7.1 nM T09572 CIC0H8 10218194 Ki = 77 nM T09572 CH7BP9 10218547 Ki = 2162 nM T09572 CX7KR8 10218604 Ki = 23 nM T09572 CB4VT6 10224210 Ki = 2.2 nM T09572 CA1YM8 10225681 IC50 = 1.995 nM T09572 C7YUF6 10226765 Ki = 0.98 nM T09572 CP25NG 10229815 Ki = 46 nM T09572 CKMB46 10230235 Ki = 26 nM T09572 C78KEN 10230490 Ki = 0.41 nM T09572 CEO3C0 10230947 Ki = 10 nM T09572 CNHR93 10231050 IC50 = 160 nM T09572 CX5S8V 10231341 Ki = 1.2 nM T09572 CT50QF 10238912 Ki = 13 nM T09572 C2AV9K 10239389 Ki = 215 nM T09572 CWTM13 10239448 Ki = 180 nM T09572 CY3B9V 10239505 Ki = 6 nM T09572 C9ZR5W 10239639 Ki = 690 nM T09572 C8GUX5 10239907 Ki = 9 nM T09572 C8R7NE 10239929 Ki = 1667 nM T09572 C2JY5L 10239930 Ki = 786 nM T09572 C4M9EA 10248906 IC50 = 30 nM T09572 CY3C6Z 10250850 IC50 = 24 nM T09572 CC94UL 10255474 IC50 = 850 nM T09572 CC7K0Q 10256914 Ki = 29 nM T09572 CRI6L0 10257135 Ki = 12 nM T09572 C9U7QP 10257298 Ki = 23 nM T09572 C46ALH 10258364 IC50 = 0.71 nM T09572 CK7W0O 10273126 Ki = 2.4 nM T09572 CM8Q4V 10274635 IC50 = 7 nM T09572 CZ7TK1 10277136 Ki = 79.43 nM T09572 C4HN5M 10277257 Ki = 398.11 nM T09572 CNY7O0 10280331 Ki = 61 nM T09572 C7GFV9 10281308 Ki = 7.2 nM T09572 CQAM65 10289494 Ki = 3 nM T09572 CD32KO 10289615 Ki = 2.5 nM T09572 C8GUV6 10295411 Ki = 63.1 nM T09572 C97VMZ 10297428 Ki = 9.2 nM T09572 CS6AF7 10298251 Ki = 1.4 nM T09572 C7JB9Z 10301472 Ki = 1.6 nM T09572 CP4MX9 10303281 Ki = 12 nM T09572 C3ZJY6 10303307 IC50 = 79 nM T09572 CA5PV1 10304239 Ki = 40 nM T09572 C16TVN 10310161 IC50 = 12 nM T09572 C2IG7F 10310316 IC50 = 2.8 nM T09572 C5NVX2 10310772 Ki = 3 nM T09572 CUZ0N7 10310778 IC50 > 4000 nM T09572 C8X2OD 10311260 Ki = 1174 nM T09572 CS5YX7 10311798 Ki = 141 nM T09572 C51CRS 10312052 Ki = 13 nM T09572 CHR1A3 10312086 Ki = 3247 nM T09572 CCRI74 10312244 Ki = 16 nM T09572 CMC1G5 10319824 IC50 = 2410 nM T09572 CQ9RL7 10325994 Ki = 36 nM T09572 CVO3N7 10344176 IC50 = 6.4 nM T09572 C3YB4P 10345121 IC50 = 1.9 nM T09572 CSB63G 10345845 IC50 = 0.46 nM T09572 CIW12H 10347752 Ki = 15 nM T09572 CHE8C4 10347753 Ki = 138 nM T09572 C3LZ7G 10347754 Ki = 13 nM T09572 CC3GW1 10348080 Ki = 15 nM T09572 C3WC2E 10348147 Ki = 54 nM T09572 C3KOI9 10348749 Ki = 24 nM T09572 C9FI8M 10360874 IC50 = 0.4 nM T09572 CQG45X 10361342 IC50 = 30 nM T09572 CMD9J2 10385550 IC50 > 100000 nM T09572 C3C2LS 10386162 IC50 = 20 nM T09572 CP4S9C 10386529 IC50 = 77 nM T09572 CAI68E 10388351 IC50 = 5 nM T09572 CF17HN 10388352 IC50 = 20 nM T09572 CL83KQ 10388797 IC50 = 16 nM T09572 C36BOF 10389430 IC50 = 63 nM T09572 CESG32 10389978 IC50 = 6.1 nM T09572 C7W4TF 10391177 IC50 = 2.7 nM T09572 C39PRE 10392311 Ki = 22 nM T09572 C5EXD4 10408758 IC50 = 149 nM T09572 CS6MA7 10413283 IC50 = 1 nM T09572 CWU0O3 10415704 Ki = 9.3 nM T09572 CYD95P 10433825 IC50 = 6 nM T09572 C6T7WB 10434776 IC50 = 50 nM T09572 CFV7D4 10436090 IC50 = 8.1 nM T09572 C2LYJ4 10436663 Ki = 26 nM T09572 CV9KC4 10436862 Ki = 138 nM T09572 C5SX2J 10443228 IC50 > 2000 nM T09572 C07KPU 10456755 IC50 = 88 nM T09572 CY17SB 10459635 IC50 = 0.71 nM T09572 CGQ62I 10460913 Ki > 1000 nM T09572 CO42XC 10461033 Ki = 16 nM T09572 CN85WI 10480652 IC50 = 3450 nM T09572 COLB47 10481477 IC50 = 1 nM T09572 C8GV3E 10483604 Ki = 119 nM T09572 CHI65E 10483729 Ki = 5100 nM T09572 CSP9I7 10483799 Ki > 1000 nM T09572 CV5GD3 10483882 Ki > 1000 nM T09572 C8SK7B 11156521 Ki = 7.3 nM T09572 CUD3I6 11156790 Ki = 14 nM T09572 C7SZD0 11165058 IC50 = 90 nM T09572 C52FBG 11166395 IC50 = 10 nM T09572 CLY23H 11168108 Ki = 16.3 nM T09572 C19UHW 11168186 Ki = 1.8 nM T09572 C6Y7LA 11168831 Ki = 1.9 nM T09572 CJ30VR 11168918 Ki = 6.7 nM T09572 C0N1BS 11169159 Ki = 21.3 nM T09572 CCA26O 11178792 IC50 = 71 nM T09572 CRW5M2 11190261 IC50 = 146 nM T09572 C9W0VG 11191034 Ki = 1.7 nM T09572 C7YZ1U 11191656 Ki = 6.8 nM T09572 CPS26T 11201645 IC50 = 0.9 nM T09572 C50SKJ 11201867 IC50 = 67 nM T09572 C24JXQ 11204090 IC50 = 83 nM T09572 C8AS3V 11211551 IC50 = 178 nM T09572 C7E9AN 11222404 IC50 = 3.3 nM T09572 CX47OL 11236807 Ki = 4.7 nM T09572 CC62PB 11238080 Ki = 2.7 nM T09572 CSPC85 11238695 Ki = 20 nM T09572 C64KCU 11238718 Ki = 1145 nM T09572 CW07ZE 11246373 IC50 = 369 nM T09572 CAS5P8 11247985 Ki = 19 nM T09572 CZ98EU 11259253 IC50 = 5 nM T09572 CIM40L 11259560 IC50 > 10000 nM T09572 CKBJ08 11260997 Ki = 8.2 nM T09572 C2U7OP 11270012 Ki = 7.4 nM T09572 CB8ZS6 11270984 IC50 = 558 nM T09572 C7JP8R 11272081 Ki = 8.4 nM T09572 CFZP19 11282448 IC50 = 287 nM T09572 CJ3Q4Y 11282697 Ki = 233 nM T09572 CCWK17 11284878 IC50 = 140 nM T09572 C49PQG 11292322 IC50 = 35 nM T09572 CCG2J7 11295707 Ki = 12.5 nM T09572 C4JK1H 11296279 IC50 = 320 nM T09572 CU4L6M 11304816 IC50 = 58 nM T09572 CP98MD 11306487 Ki = 98 nM T09572 CN38VE 11307645 Ki = 1.5 nM T09572 CK9E2Y 11317465 Ki = 20 nM T09572 CK4P6A 11317824 Ki = 20.7 nM T09572 CO7CX6 11318577 Ki = 391 nM T09572 CCU9P8 11318709 Ki = 39 nM T09572 CWT28O 11328029 IC50 = 6 nM T09572 C7R2ZE 11329623 Ki = 5.6 nM T09572 C47VRG 11329860 Ki = 6.2 nM T09572 CR1BG6 11330800 Ki = 3000 nM T09572 CZ6FG9 11340348 Ki = 3.1 nM T09572 C5R2GO 11340894 Ki = 139 nM T09572 CR1K5W 11342160 IC50 = 250 nM T09572 CVGM47 11351174 IC50 = 78 nM T09572 CHJ73G 11353174 Ki = 2.2 nM T09572 C36OES 11374857 IC50 = 160 nM T09572 C43HJQ 11376081 Ki = 4 nM T09572 CQ58NT 11376122 Ki = 27 nM T09572 CU3V1H 11387603 Ki = 197 nM T09572 C3XR6W 11408441 IC50 = 5 nM T09572 C7MVN8 11409615 Ki = 70.8 nM T09572 CBL42Y 11410080 Ki = 327.6 nM T09572 CI8X2J 11410430 Ki = 25.7 nM T09572 CI80HK 11410594 Ki = 405 nM T09572 CF6XZ1 11419337 IC50 = 12 nM T09572 C2RXD8 11419338 IC50 = 46 nM T09572 C0EHV3 11419666 IC50 = 24.5 nM T09572 CI3RU9 11419776 IC50 = 15 nM T09572 C26DPU 11420203 Ki = 7.1 nM T09572 C28YHB 11420543 Ki = 11 nM T09572 C69OFJ 11420621 Ki = 5.8 nM T09572 CB51KQ 11433168 Ki = 26 nM T09572 CXY0L4 11442761 IC50 = 4 nM T09572 CTAI65 11452967 Ki = 6 nM T09572 CJP2I6 11453830 IC50 = 1985 nM T09572 C09HMW 11454965 Ki = 4.9 nM T09572 C50BVO 11455871 Ki = 4.9 nM T09572 CKU5J7 11464405 IC50 = 4 nM T09572 C5JFE2 11467626 Ki = 14.2 nM T09572 CN54JD 11476556 IC50 = 772000 nM T09572 CI6CY2 11489130 Ki = 8.9 nM T09572 C1I3TF 11489588 Ki = 13.7 nM T09572 CMQ86R 11495432 IC50 = 5 nM T09572 C6L8DU 11495754 IC50 = 2.1 nM T09572 C9YME5 11496313 IC50 = 1.6 nM T09572 CZG39V 11496739 IC50 = 2.3 nM T09572 CQF0N9 11496824 Ki = 92 nM T09572 CE0FW1 11497179 Ki = 15 nM T09572 CSG7A1 11497180 Ki = 87 nM T09572 CZIE58 11502008 IC50 = 5.8 nM T09572 COC9S1 11504274 IC50 = 6 nM T09572 CEGY35 11504793 Ki = 180 nM T09572 CRVH23 11504906 Ki = 2.8 nM T09572 C10FVQ 11505089 IC50 = 13 nM T09572 CCP2Z0 11510399 IC50 = 4 nM T09572 CB59MV 11510669 IC50 = 145 nM T09572 C72BCW 11510887 IC50 = 266 nM T09572 CTKH79 11511219 IC50 = 25 nM T09572 CW6C2K 11511638 Ki = 2190 nM T09572 CXH3M7 11511671 Ki = 9.6 nM T09572 C9DE5V 11511776 IC50 = 15 nM T09572 C2B6YR 11512135 IC50 = 5.9 nM T09572 CVW89A 11512221 Ki = 6.6 nM T09572 CEPN59 11516903 IC50 = 45 nM T09572 C7O3YC 11517116 IC50 > 1000 nM T09572 CKH3R6 11518999 Ki = 3.3 nM T09572 CI1H6G 11519341 Ki > 3000 nM T09572 CW4V9C 11519451 Ki = 1.8 nM T09572 CZN1S8 11519652 Ki = 3000 nM T09572 CB86YA 11525369 IC50 = 57 nM T09572 C1TLH5 11526309 IC50 = 78 nM T09572 CGU14V 11526592 Ki = 30 nM T09572 CMCE20 11526824 IC50 = 93 nM T09572 CL04IY 11527169 Ki = 44 nM T09572 CQ7LC4 11531010 IC50 = 8 nM T09572 C24VTF 11531660 IC50 = 41 nM T09572 C4W2IN 11533195 IC50 = 35 nM T09572 C8W1XB 11533835 Ki = 8 nM T09572 CQ08DH 11539632 IC50 = 85 nM T09572 C5NA7O 11541231 Ki = 1615 nM T09572 C3E9MH 11545677 IC50 = 9 nM T09572 CP8I4R 11546687 IC50 = 734 nM T09572 CI15ZK 11547011 Ki = 3.3 nM T09572 CE34IS 11547939 IC50 = 9.7 nM T09572 CX6IL5 11548234 IC50 = 1.5 nM T09572 C69YGT 11548597 Ki = 3.5 nM T09572 C0KYZ7 11553316 IC50 = 163 nM T09572 CW4QS9 11553648 IC50 = 150 nM T09572 C0I6EV 11553871 IC50 = 1.585 nM T09572 CZD24Q 11554412 IC50 = 3 nM T09572 CPM70L 11554989 IC50 = 48 nM T09572 C64NID 11555572 IC50 = 37 nM T09572 CNWU65 11556070 IC50 = 2 nM T09572 C5WKO2 11559625 IC50 = 18 nM T09572 C7J9IY 11560917 IC50 = 6 nM T09572 CXR53E 11561126 IC50 = 0.5 nM T09572 C0XQ1U 11561155 IC50 = 120 nM T09572 CS5M0K 11562056 Ki = 52 nM T09572 CF8E0C 11562129 IC50 = 100 nM T09572 CDP1L5 11562138 IC50 = 2 nM T09572 CX3HC8 11563017 IC50 = 11 nM T09572 CY0N7L 11563153 IC50 = 340 nM T09572 C59SVL 11563383 IC50 = 21 nM T09572 CMFZ35 11568741 IC50 = 339 nM T09572 C2BIP8 11568782 IC50 = 29 nM T09572 C0J3VR 11569300 IC50 = 32 nM T09572 CAEY52 11569327 Ki = 2 nM T09572 CAC92H 11569340 IC50 = 302 nM T09572 CN0S1H 11570031 IC50 = 31 nM T09572 CJ9RX4 11570040 Ki = 3.5 nM T09572 C8FXD6 11577410 Ki = 2.3 nM T09572 CN87ZF 11577588 IC50 = 22 nM T09572 C2YIV1 11577708 Ki = 727 nM T09572 CXKA03 11581666 IC50 = 3628 nM T09572 CM0H2R 11583049 IC50 = 2 nM T09572 CZ6C8H 11583193 IC50 = 1 nM T09572 CPA3J7 11583744 IC50 = 2.7 nM T09572 CNT0J4 11583747 IC50 = 2 nM T09572 CP07QN 11583835 IC50 = 20 nM T09572 C70NAD 11583925 IC50 = 330 nM T09572 CS6OE5 11584710 Ki = 2.5 nM T09572 COE14C 11589812 IC50 = 38 nM T09572 CNB39X 11591169 IC50 = 50 nM T09572 C5SOE3 11591542 IC50 = 380 nM T09572 CLW26H 11591644 IC50 = 8 nM T09572 CD6Y3F 11592099 IC50 = 2 nM T09572 C3E9YV 11592199 IC50 = 88 nM T09572 CLEA14 11592317 Ki = 129 nM T09572 CMAF85 11596311 IC50 = 6.6 nM T09572 CAU85E 11597758 IC50 = 313 nM T09572 C9OU8J 11598355 IC50 = 2 nM T09572 CE0N5F 11599186 IC50 = 16 nM T09572 C0H3WV 11599681 IC50 = 5360 nM T09572 CKI9D5 11599973 IC50 = 6 nM T09572 CS1EL0 11603897 IC50 = 7 nM T09572 CRAO19 11604236 IC50 = 297 nM T09572 CCL5H9 11605260 IC50 = 1050 nM T09572 C97GBU 11605775 IC50 = 49 nM T09572 CEF85Q 11605821 Ki = 11 nM T09572 CC5R1Q 11610423 Ki = 2.3 nM T09572 CP4VN0 11611530 IC50 = 60 nM T09572 C9I5GN 11612098 IC50 = 19 nM T09572 CYB0H4 11612847 Ki = 190 nM T09572 CM03ZX 11613073 IC50 = 1.7 nM T09572 CDA48G 11613696 Ki = 3.7 nM T09572 CP9T8V 11613829 Ki = 9.3 nM T09572 CG1RP5 11619850 IC50 = 3 nM T09572 CDT2Y7 11620005 IC50 = 540 nM T09572 CIO53A 11627085 IC50 = 44 nM T09572 C2NC0H 11627122 IC50 = 9 nM T09572 CHS10O 11627316 Ki = 13 nM T09572 CGEX14 11627530 IC50 = 1.3 nM T09572 C3CI5V 11627700 Ki = 6 nM T09572 CVA6R9 11628136 Ki = 41 nM T09572 CEK0Z8 11628328 IC50 = 25 nM T09572 C6CXP5 11628547 Ki = 221 nM T09572 CA90RE 11632484 IC50 = 20 nM T09572 C7H9VD 11632909 IC50 = 461 nM T09572 CCN9E6 11633862 IC50 = 90 nM T09572 CE70ZA 11634061 IC50 = 42 nM T09572 CX36IC 11634230 IC50 = 98 nM T09572 CP46KM 11634329 Ki = 13 nM T09572 CBW24J 11634823 IC50 = 38 nM T09572 C75FNR 11634886 IC50 = 26 nM T09572 CDE1G8 11635187 IC50 = 25 nM T09572 C8Y9AL 11635230 IC50 = 99 nM T09572 C8LU4M 11635274 Ki = 4.8 nM T09572 CUN3R9 11635332 IC50 = 74 nM T09572 C0PQ9D 11635674 Ki = 1.8 nM T09572 C5U4HW 11635715 Ki = 67 nM T09572 CY3IN5 11640515 IC50 = 24 nM T09572 C8SBV2 11641333 Ki = 605 nM T09572 CH79OL 11641948 IC50 = 15 nM T09572 CUG36W 11642443 Ki = 37 nM T09572 CLFC12 11642491 Ki = 96 nM T09572 CKM2Z4 11646818 IC50 = 10 nM T09572 CJQK24 11647458 IC50 = 10 nM T09572 C5A4YW 11648240 IC50 = 13 nM T09572 CTLK95 11648753 Ki = 8.9 nM T09572 CK2SO9 11648912 IC50 = 0.1 nM T09572 C1XZ5S 11648976 Ki = 161 nM T09572 C0WAT8 11649549 IC50 = 3 nM T09572 CE57QF 11653882 IC50 = 20 nM T09572 C8I7UT 11654412 IC50 = 5.6 nM T09572 CM0J9D 11654904 IC50 > 1000 nM T09572 CRF2O3 11655701 Ki = 18 nM T09572 CFHR60 11655790 IC50 > 1000 nM T09572 CP09GF 11655872 IC50 = 29 nM T09572 CTW7H9 11656044 IC50 = 151 nM T09572 CI3YO9 11656489 IC50 = 29 nM T09572 C35CMI 11656728 Ki = 1300 nM T09572 CT0YF3 11656805 Ki = 160 nM T09572 C2TDF5 11656916 Ki = 71.4 nM T09572 C6Q7TC 11657090 Ki = 22 nM T09572 CJ8OS7 11662564 IC50 = 158 nM T09572 C1F9VA 11662657 IC50 = 4 nM T09572 CESA67 11662906 IC50 = 22 nM T09572 CZ0KM9 11663109 IC50 > 1000 nM T09572 C91WGJ 11664086 Ki = 32 nM T09572 CW0C5S 11664134 Ki = 3000 nM T09572 C5NI1G 11670645 Ki = 648 nM T09572 CMXQ27 11671178 Ki = 2.9 nM T09572 CX3WF2 11676200 IC50 = 710 nM T09572 CXB59V 11676220 IC50 = 1.4 nM T09572 C0R5KF 11677277 IC50 = 2 nM T09572 CW1MI7 11677806 IC50 = 109 nM T09572 CW0N1P 11678040 Ki = 4.4 nM T09572 C4KG5D 11678370 IC50 = 140 nM T09572 C8UVK4 11678666 Ki = 394 nM T09572 CD7C4O 11683259 IC50 = 5.4 nM T09572 CEHG64 11683903 IC50 = 16 nM T09572 CG76YZ 11684745 IC50 = 45 nM T09572 C8S2RG 11691468 Ki = 16.98 nM T09572 CR0JZ3 11691995 IC50 = 54 nM T09572 C8CWF4 11692133 Ki = 7 nM T09572 CKX65Z 11692293 IC50 = 519 nM T09572 C3HOB4 11692382 Ki = 167 nM T09572 CJ6C2T 11692643 Ki = 29 nM T09572 C6QKV2 11698276 Ki = 380 nM T09572 C17ZOJ 11698592 Ki = 3.6 nM T09572 CW5Z4U 11698729 Ki = 340 nM T09572 C3D1IX 11698964 Ki = 33 nM T09572 CMZ94P 11699265 Ki = 15 nM T09572 CYR87W 11705240 IC50 = 19 nM T09572 CR6BE5 11705485 IC50 = 29 nM T09572 CG2LE3 11706442 IC50 = 39 nM T09572 CE1FU8 11706443 IC50 = 41 nM T09572 C16BRA 11706744 Ki = 4 nM T09572 CKZJ72 11710969 IC50 > 1000 nM T09572 CIZQ65 11711452 IC50 = 7 nM T09572 CL3H6E 11712583 IC50 = 39 nM T09572 C8V9XO 11712898 IC50 = 29 nM T09572 C1MV6S 11713027 IC50 = 1.4 nM T09572 CWQ67V 11713742 IC50 = 23 nM T09572 C74DRE 11719291 IC50 = 7 nM T09572 C87WCU 11719447 Ki = 1 nM T09572 CIR3H9 11719877 Ki = 8.2 nM T09572 CO29BN 11719912 IC50 = 39 nM T09572 CQV4D8 11720881 Ki = 61 nM T09572 C3CSB2 11740891 IC50 = 26 nM T09572 CG70PF 11743571 IC50 = 2 nM T09572 C7IR0M 11752320 IC50 = 5.2 nM T09572 CFB78R 11752339 Ki = 7.9 nM T09572 C6T9RV 11752579 Ki = 7.1 nM T09572 CIB4J8 11752750 Ki = 3 nM T09572 C0REU4 11756387 Ki = 38 nM T09572 C8KZ7Y 11758076 Ki = 11 nM T09572 C15NMU 11758499 Ki = 9.7 nM T09572 CDT5W6 11775399 IC50 = 1.4 nM T09572 C7JD4S 11775505 IC50 = 71 nM T09572 CMT60I 11778029 IC50 = 310 nM T09572 CX20YM 11785261 Ki = 9.2 nM T09572 CJZ1S6 11785262 Ki = 8.8 nM T09572 C3URN6 11785761 Ki = 11.4 nM T09572 CCA5X9 11786179 Ki = 374 nM T09572 CF5X6S 11786476 Ki = 166 nM T09572 CQ3UA0 11837128 IC50 = 191 nM T09572 C8MT6W 11973798 IC50 = 427 nM T09572 CA54WB 11973799 IC50 = 13 nM T09572 C09SBY 11973800 IC50 = 966 nM T09572 C4G3JS 11973801 IC50 = 53 nM T09572 CJ51DI 11973802 IC50 = 1690 nM T09572 CW4V0D 11973803 IC50 > 2000 nM T09572 C0X9SH 11973913 IC50 > 2000 nM T09572 CY6F0Q 11973915 IC50 > 2000 nM T09572 CYA98F 11973916 IC50 = 1140 nM T09572 CTQ2M5 11974030 IC50 = 178 nM T09572 C9OQ1D 11974034 IC50 = 351 nM T09572 C1NEZ7 11974035 IC50 = 187 nM T09572 CRP64S 11974126 IC50 = 132 nM T09572 CYF81E 11974128 IC50 > 2000 nM T09572 C68TIS 11974129 IC50 = 1480 nM T09572 CU3J7M 11974130 IC50 = 59 nM T09572 CN38YH 11974131 IC50 = 137 nM T09572 C05LEI 11974132 IC50 = 393 nM T09572 C72WDJ 11974227 IC50 = 99 nM T09572 C1BXQ6 11974228 IC50 = 418 nM T09572 C5W7EA 11974229 IC50 = 601 nM T09572 C3C2EN 11974230 IC50 = 171 nM T09572 CAN81B 11974231 IC50 = 31 nM T09572 C2QW4A 11974233 IC50 = 2150 nM T09572 CHJ84N 11974345 IC50 = 159 nM T09572 CNCP71 11974346 IC50 = 39 nM T09572 C7W6UZ 11975326 IC50 = 192 nM T09572 CJ82RK 11975327 IC50 = 24 nM T09572 C8KJU9 11975436 IC50 = 75 nM T09572 C3EU8T 11975438 IC50 = 60 nM T09572 CJ0M5S 11975440 IC50 > 700 nM T09572 CGHS90 11993892 IC50 = 2 nM T09572 CC67HK 11993893 IC50 = 0.89 nM T09572 CY2R0H 11993894 IC50 = 1.3 nM T09572 CTR36W 11993895 IC50 = 6.1 nM T09572 CH46NZ 11993896 IC50 = 6.2 nM T09572 CY93VJ 11993897 IC50 = 37 nM T09572 CKJ40R 11994017 IC50 = 3.2 nM T09572 C2X1FE 11994018 IC50 = 6918 nM T09572 COYJ12 11994019 IC50 = 3.4 nM T09572 C2XV4Y 11994136 IC50 = 8.5 nM T09572 CZO24Q 11994137 IC50 = 25 nM T09572 CU4ZI8 11994138 IC50 = 24 nM T09572 CE0D8U 11994273 IC50 > 10000 nM T09572 C87MRI 11994275 IC50 = 31.6 nM T09572 CUT45B 11994276 IC50 > 10000 nM T09572 CO9RD2 11994277 IC50 = 5 nM T09572 CB47ZX 11994412 IC50 = 0.87 nM T09572 C2TXD4 11994413 IC50 = 1.1 nM T09572 C1FLA4 11994414 IC50 = 3.1 nM T09572 CP3ID2 11994659 IC50 = 1.3 nM T09572 CX49YR 11994660 IC50 = 2.5 nM T09572 C8WS7J 11994661 IC50 = 5.7 nM T09572 CID9L3 11994662 IC50 = 29 nM T09572 CNOW76 11994780 IC50 = 1.4 nM T09572 CKS43A 11994784 IC50 = 1.1 nM T09572 C75HYU 11994786 IC50 = 1.1 nM T09572 CXJ16Z 11994909 IC50 > 10000 nM T09572 C79ATS 11994910 IC50 = 1412 nM T09572 C9SDQ6 11994911 IC50 = 2.7 nM T09572 CGJD13 11994912 IC50 = 0.75 nM T09572 CH52LD 11994913 IC50 = 1.3 nM T09572 CDI85R 11995024 IC50 = 0.91 nM T09572 CB8E2J 11995025 IC50 = 2 nM T09572 C1F3KB 11995026 IC50 = 38 nM T09572 CL8U5H 11995028 IC50 = 9.5 nM T09572 CUTI13 11995136 IC50 = 794 nM T09572 C6X5QK 11995137 IC50 = 3980 nM T09572 C7CQ0R 11995138 IC50 = 40 nM T09572 C65FGL 11995139 IC50 = 478 nM T09572 CO3S6Y 11995140 IC50 = 36 nM T09572 CUG9Q0 11995141 IC50 = 200 nM T09572 CA0TX2 11995240 IC50 = 63 nM T09572 CM12WP 11995241 IC50 = 87 nM T09572 C7VYA1 11995242 IC50 = 1 nM T09572 C6AT2K 11995243 IC50 = 5.6 nM T09572 C48VEJ 11995244 IC50 = 1.5 nM T09572 C5RE4A 11995245 IC50 = 3.1 nM T09572 C56OSH 11995342 IC50 = 3.1 nM T09572 CV28MQ 11995343 IC50 = 19 nM T09572 C19YGN 11995344 IC50 = 3.8 nM T09572 C9L5UO 11995345 IC50 = 3.5 nM T09572 CR8C7Y 11995346 IC50 = 4168 nM T09572 CDV83P 11995347 IC50 = 2.3 nM T09572 COUR13 11995441 IC50 = 5.3 nM T09572 CZ23MA 11995442 IC50 = 3.5 nM T09572 C91ZIU 11995443 IC50 = 7.7 nM T09572 CKF0H1 11995444 IC50 = 3.2 nM T09572 CG9Z2R 11995445 IC50 = 7 nM T09572 C0QSD9 11995552 IC50 = 4.9 nM T09572 CY07CV 11995644 IC50 = 1258 nM T09572 CZQ39K 11995645 IC50 = 501 nM T09572 CE2OQ3 11995646 IC50 = 31 nM T09572 C41NIS 11995647 IC50 = 501 nM T09572 CSJ72B 11995648 IC50 = 0.74 nM T09572 CM6P0A 12002494 IC50 > 5000 nM T09572 CZ0UY2 12020149 Ki = 20 nM T09572 C9L6BY 12020151 IC50 = 100 nM T09572 CR64CY 12020152 Ki = 51 nM T09572 C42JBR 12020156 IC50 = 270 nM T09572 C61WZV 12020161 Ki = 108 nM T09572 CLP70H 12020164 Ki = 191 nM T09572 CN3FB9 12020168 Ki = 795 nM T09572 CICW40 12020169 Ki = 266 nM T09572 CY6BQ4 15133403 EC50 = 140 nM T09572 C7WB4Y 15981934 Ki > 5000 nM T09572 CL50KS 15983730 Ki = 220 nM T09572 CD39IP 15983731 Ki > 5000 nM T09572 CM1I3Z 15983732 Ki > 5000 nM T09572 C4QLI2 15983733 Ki = 341 nM T09572 CGUZ74 15983734 Ki > 5000 nM T09572 C8PFB1 15983862 Ki = 357 nM T09572 C9A0LX 15983863 Ki > 5000 nM T09572 C76FSJ 15983864 Ki = 707 nM T09572 CDT5B7 15983865 Ki = 2060 nM T09572 C43HRS 15983866 Ki > 5000 nM T09572 CXW37K 15987265 IC50 = 5 nM T09572 CQ2H5X 15987638 IC50 = 2630 nM T09572 C8FV4Y 16006976 Ki = 6 nM T09572 CL2PB7 16006977 Ki = 7 nM T09572 CKJ76E 16006978 IC50 = 2.2 nM T09572 CB0JD2 16037921 Ki = 1 nM T09572 CX9W7Q 16043220 Ki = 21 nM T09572 CFM31I 16043291 Ki = 0.6 nM T09572 CB6LK8 16046114 Ki = 19.95 nM T09572 CR78OW 16046124 Ki = 3.981 nM T09572 CD65KI 16046157 Ki = 51 nM T09572 CA5YN3 16049789 IC50 = 0.3 nM T09572 C3LK2C 16072132 Ki = 3 nM T09572 CRU35S 16106513 Ki = 77 nM T09572 CJ4M0E 16110074 Ki = 31.62 nM T09572 CU37CY 16116777 Ki = 39.81 nM T09572 CJLX24 16192241 IC50 = 11000 nM T09572 C72BAI 16659061 Ki = 78 nM T09572 C23NUI 16659197 Ki = 140 nM T09572 COC0B8 16659239 Ki = 16000 nM T09572 CYS2H0 16659240 IC50 = 20 nM T09572 CFXU61 16718619 IC50 = 13 nM T09572 C7K5AW 16721015 IC50 = 1 nM T09572 CV5F3P 16739263 IC50 = 29 nM T09572 CO1W7Z 16739310 Ki = 8 nM T09572 CTB2D8 16739324 Ki = 10 nM T09572 CGCY91 16742745 IC50 = 154 nM T09572 C2IJ3D 16742746 IC50 = 7 nM T09572 C4URY2 16742747 IC50 = 20 nM T09572 C8V1KM 16745235 IC50 = 3 nM T09572 CDK04H 16745305 Ki = 43 nM T09572 C96RYO 17173466 IC50 = 23000 nM T09572 COL97Q 17484866 IC50 = 6500 nM T09572 C7HA3N 17545006 IC50 = 23000 nM T09572 C5SO0V 17848895 IC50 = 190 nM T09572 CSTQ69 17989325 Ki = 398.11 nM T09572 CJ7Z4X 17989329 Ki = 19.95 nM T09572 CWC4K6 17989356 Ki = 125.89 nM T09572 CL2QF0 17989369 Ki = 15.85 nM T09572 CYV93L 17989373 Ki = 50.12 nM T09572 C5P3IU 17989383 Ki = 316.23 nM T09572 CKX23J 17989406 Ki = 31.62 nM T09572 C5X4FZ 17989409 Ki = 25 nM T09572 C6SZ0G 17989439 Ki = 82 nM T09572 CVSB32 18361509 IC50 > 1000 nM T09572 CI46GT 18435902 IC50 = 1.8 nM T09572 C2DFS4 18435980 IC50 = 6.6 nM T09572 C03YQS 18435984 IC50 = 35 nM T09572 CQ86SW 18435986 IC50 = 48 nM T09572 C0IPE3 18435988 IC50 = 23 nM T09572 CFYX59 18436038 IC50 = 2 nM T09572 C37CPM 18436043 IC50 = 1600 nM T09572 CCS6E4 18436055 IC50 = 0.74 nM T09572 C7MUE8 18436066 IC50 = 0.36 nM T09572 C9HN3G 18436075 IC50 = 9.2 nM T09572 CA9UL8 18436082 IC50 = 1.4 nM T09572 CDQS35 18436083 IC50 = 1.4 nM T09572 C1WJ0Z 18436085 IC50 = 10 nM T09572 C3CYE7 18436094 IC50 = 0.92 nM T09572 C56SPK 18436095 IC50 = 110 nM T09572 C5Z8FL 18436109 IC50 = 170 nM T09572 CF7Q1R 18436112 IC50 = 3.7 nM T09572 CS24AR 18436114 IC50 = 0.53 nM T09572 C34WKZ 18436115 IC50 = 2.2 nM T09572 C0H7OP 18436117 IC50 = 1 nM T09572 CXL27Y 18436118 IC50 = 100 nM T09572 C0ST8U 18436119 IC50 = 3.2 nM T09572 C7X1SY 18436120 IC50 = 4.1 nM T09572 C9F2DA 18436123 IC50 = 25 nM T09572 C32IMY 18436125 IC50 = 26 nM T09572 CW6HU8 18436126 IC50 = 18 nM T09572 CCN82B 18436129 IC50 = 73 nM T09572 CAP6L1 18672590 Ki = 31.62 nM T09572 CBR6Q7 20608969 Ki = 61 nM T09572 COF9E8 20608974 Ki = 19 nM T09572 CWSB30 20608975 Ki = 13 nM T09572 C7PL9M 20608976 Ki = 42 nM T09572 CG9R3I 20608977 Ki = 40 nM T09572 C9U6JQ 20608981 Ki = 8 nM T09572 CC1RB9 20608989 Ki = 190 nM T09572 C2H1YF 20608991 Ki = 25 nM T09572 C8Q0XO 20608992 Ki = 45 nM T09572 C8CUT0 20608996 Ki = 249 nM T09572 CVGY56 20609011 Ki = 63 nM T09572 C7N6XY 20609018 Ki = 30 nM T09572 C78UWI 20609028 Ki = 128 nM T09572 C2PF3N 20779393 Ki = 11 nM T09572 C3QGN7 20779413 Ki = 11 nM T09572 C1R4BJ 20779426 Ki = 300 nM T09572 C84VKA 20779429 Ki = 39 nM T09572 C9NK0T 20779441 Ki = 155 nM T09572 CW81IR 20779442 Ki = 281 nM T09572 CSV2M0 20817761 IC50 = 4 nM T09572 C85YPN 20817762 IC50 = 24 nM T09572 CO29QJ 20817763 IC50 = 16 nM T09572 C7X4ND 20817800 IC50 = 44 nM T09572 CS4AU1 20817821 IC50 = 5 nM T09572 CZC89U 20817846 IC50 = 88 nM T09572 CHB01Q 20817864 IC50 = 97 nM T09572 CGP04L 20877140 Ki = 20900 nM T09572 C9OMT8 21062990 IC50 = 65 nM T09572 CD90IG 21062991 IC50 = 140 nM T09572 CTCV19 21062998 IC50 = 7.4 nM T09572 CXC0F1 21062999 IC50 = 11 nM T09572 C01EQU 21063019 IC50 > 10000 nM T09572 C89XCE 21063022 IC50 > 1000 nM T09572 CJRD60 21101400 Ki = 39.81 nM T09572 CSU46X 21101402 Ki = 25.12 nM T09572 CXA8V1 21101416 Ki = 1000 nM T09572 CHZ4L6 21108056 IC50 = 11 nM T09572 CVS4D7 21108099 IC50 = 100 nM T09572 CD3O2Y 21108114 IC50 = 34 nM T09572 CYU8L1 21108117 IC50 = 20 nM T09572 C8R7XC 21108118 IC50 = 30 nM T09572 C48PMV 21939767 IC50 = 91 nM T09572 CIS5W2 21939881 IC50 = 230 nM T09572 CZ1GI7 21939887 IC50 = 350 nM T09572 CLD4C5 21939898 IC50 = 1.6 nM T09572 CC98QY 21939900 IC50 = 10000 nM T09572 CFS7G5 21939902 IC50 = 2.8 nM T09572 CDKT72 21939915 IC50 = 8.4 nM T09572 C4R6QP 21939935 IC50 = 380 nM T09572 CG63ZA 21939937 IC50 = 1.4 nM T09572 CI9R2D 21939940 IC50 = 380 nM T09572 CD8GZ7 21939950 IC50 = 2.2 nM T09572 CU7Z2B 21940008 IC50 = 17 nM T09572 C12GZE 21940052 IC50 = 190 nM T09572 CBQV01 21940083 IC50 = 1.9 nM T09572 C1MD6T 22018856 IC50 = 2 nM T09572 CK0GB9 22018896 IC50 = 12 nM T09572 CBO1J2 22018914 IC50 = 5 nM T09572 C0FJO5 22018919 IC50 = 10 nM T09572 CZUW58 22018932 IC50 = 5 nM T09572 C92HPN 22018944 IC50 = 1 nM T09572 C5SG9E 22018945 IC50 = 2 nM T09572 C2FYN1 22018957 IC50 = 0.5 nM T09572 CSQ1H0 22018964 IC50 = 1 nM T09572 CCQ6M7 22018997 IC50 = 6 nM T09572 CTQG86 22018999 IC50 = 2 nM T09572 C10MAZ 22251624 IC50 = 1.8 nM T09572 CY2PZ8 22254547 IC50 > 10000 nM T09572 C0G7FB 22254553 IC50 > 2000 nM T09572 CV64TI 22254570 IC50 = 808 nM T09572 COW3D8 22254571 IC50 = 137 nM T09572 CAL1Q8 22254581 IC50 = 60 nM T09572 CTH7J3 22254632 IC50 = 115 nM T09572 C16HAP 22348022 IC50 = 1.1 nM T09572 CCU37W 22348066 IC50 = 15 nM T09572 C82XIL 22348140 IC50 = 0.8 nM T09572 CY0WA7 22348155 IC50 = 1.2 nM T09572 C5PS4N 22348219 IC50 = 34 nM T09572 C6KJ0C 22348261 IC50 = 3 nM T09572 CJ67AV 22421739 IC50 = 6600 nM T09572 CITM21 22421741 IC50 = 727000 nM T09572 CO8AL0 22421743 IC50 = 251 nM T09572 CY39TI 22421749 IC50 = 230 nM T09572 C6TDY7 22421750 IC50 = 24800 nM T09572 C5UX4T 22422406 IC50 = 250 nM T09572 CTH09W 22427041 IC50 = 327 nM T09572 CLA5H0 23022394 IC50 = 32 nM T09572 CJ86XR 23022422 IC50 = 1.8 nM T09572 C26ESM 23022499 IC50 = 13 nM T09572 CT13GQ 23022509 IC50 = 4.3 nM T09572 C46HAR 23022536 IC50 = 1.7 nM T09572 CJS4U2 23022589 IC50 = 100 nM T09572 C81XUE 23027035 IC50 = 13 nM T09572 C5LCB2 23027181 IC50 = 58 nM T09572 CR5H1I 23027211 IC50 = 4.8 nM T09572 CC2L1B 23027245 IC50 = 16 nM T09572 CQ45SO 23027402 IC50 = 6.5 nM T09572 CG9M4Y 23027411 IC50 = 10 nM T09572 CC6R2O 23027527 IC50 = 6 nM T09572 CB4TK6 23027679 IC50 = 2.5 nM T09572 CLBE26 23027806 IC50 = 2.3 nM T09572 CW86DG 23027830 IC50 = 25 nM T09572 C9S3NP 23120512 IC50 = 4.4 nM T09572 C4Z9DB 23120540 IC50 = 1000 nM T09572 CJC1Y9 23120543 IC50 > 1000 nM T09572 C40PSL 23120550 IC50 = 2.5 nM T09572 CEH84I 23120564 IC50 = 4.8 nM T09572 C01LMH 23120572 IC50 = 2 nM T09572 C14ABC 23120575 IC50 = 6.8 nM T09572 C5RY1K 23120576 IC50 = 5.6 nM T09572 CV5ES9 23120580 IC50 = 17 nM T09572 CF67MJ 23120582 IC50 = 11 nM T09572 CYM4Q8 23120586 IC50 = 4 nM T09572 CK8Y2C 23532172 IC50 = 580 nM T09572 C1JOZ3 23532179 IC50 = 100 nM T09572 CJ6O3B 23532180 IC50 = 50 nM T09572 C45MIS 23532181 IC50 = 20 nM T09572 C3P9AQ 23567276 Ki = 240 nM T09572 CYQ35D 23567283 Ki = 130 nM T09572 CVO89E 23567290 Ki = 280 nM T09572 C9CRK8 23567310 Ki = 1641 nM T09572 C8OK2Q 23567355 Ki = 122 nM T09572 CK71DM 23567391 Ki = 205 nM T09572 CV5LK9 23567394 Ki = 1080 nM T09572 C7GP0L 23567408 Ki = 300 nM T09572 C0Q8AU 23567432 Ki = 1223 nM T09572 CL9B6S 23567477 Ki = 135 nM T09572 CX7QH0 23567513 Ki = 100 nM T09572 C2DIJ7 23573799 Ki = 21 nM T09572 CKXV10 23593464 IC50 = 3.4 nM T09572 C6L9NA 23593468 IC50 = 19 nM T09572 CNSZ98 23593471 IC50 = 1300 nM T09572 CO1D9V 23593472 IC50 = 220 nM T09572 C7R5TE 23593474 IC50 = 18 nM T09572 CQ80SP 23626228 Ki = 107 nM T09572 CX7B9D 23657037 IC50 = 29 nM T09572 CGI6M2 23658492 IC50 = 45.71 nM T09572 C4C3HR 24780883 IC50 = 4.4 nM T09572 CH15KN 24808474 IC50 = 3 nM T09572 C59IBZ 24857597 Ki = 9.7 nM T09572 CB4LY1 24857598 Ki = 2.6 nM T09572 C56KFT 24952055 EC50 = 60 nM T09572 C8TB2K 24952056 EC50 = 40 nM T09572 C2L9DI 24952417 EC50 = 20 nM T09572 C2GAX4 24952418 IC50 = 13 nM T09572 CX5QB0 24952419 EC50 = 20 nM T09572 C40XUR 24952765 IC50 = 3 nM T09572 CX83WL 24963343 Ki = 6 nM T09572 CD1AO6 25017033 Ki = 5.2 nM T09572 C1HK0Y 25017297 Ki = 38 nM T09572 CE7UZ8 25017298 Ki = 14 nM T09572 C9Y2LZ 25017299 Ki = 48 nM T09572 CIL04A 25017300 Ki = 28 nM T09572 CIL0E6 25017571 Ki = 4.2 nM T09572 C8FE1I 25017572 Ki = 6.1 nM T09572 C9X5AB 25018073 Ki = 59 nM T09572 C7ZR3G 25018075 Ki = 1679 nM T09572 CHQ86P 25054013 Ki = 3.1 nM T09572 C7EQ5T 25054288 Ki = 4.7 nM T09572 CCEY27 25054289 Ki = 11.2 nM T09572 C0PIZ8 25054550 Ki = 17.3 nM T09572 C20JHU 25054551 Ki = 33 nM T09572 CG8C7J 25054804 Ki = 12 nM T09572 C2FP5D 25056872 Ki = 24.3 nM T09572 C6Z3CE 25057124 Ki = 22.6 nM T09572 C0TYE6 25057388 Ki = 4.7 nM T09572 CE12CD 25057645 Ki = 43.4 nM T09572 C1K9VQ 25057911 Ki = 9.4 nM T09572 CH4PI7 25057913 Ki = 30.4 nM T09572 C8L6JE 25058425 IC50 = 1 nM T09572 C9WI7E 25110804 Ki = 3 nM T09572 CWVK74 25113835 IC50 = 3 nM T09572 CZH60W 25113838 IC50 = 8 nM T09572 CN8XF7 25114064 IC50 = 42 nM T09572 C9XL7R 25114065 IC50 = 56 nM T09572 CU10OY 25114067 IC50 = 4 nM T09572 CCQE40 25114068 IC50 = 16 nM T09572 CAW76X 25114286 IC50 = 1 nM T09572 CPD2X6 25114287 IC50 = 4 nM T09572 CCN5Y9 25114722 IC50 = 5 nM T09572 CCF8W5 25114723 IC50 = 19 nM T09572 CN5F7X 25114724 IC50 = 213 nM T09572 CS85TU 25114948 IC50 = 300 nM T09572 C38NAY 25115173 IC50 = 32 nM T09572 CPU90J 25115618 IC50 = 2 nM T09572 C9PQR0 25115619 IC50 = 10000 nM T09572 CT61UB 25115621 IC50 = 29 nM T09572 C1U6ES 25115852 IC50 = 74 nM T09572 CQLV30 25115854 IC50 = 10 nM T09572 CQ2U9N 25115855 IC50 = 5 nM T09572 C9V8QS 25115856 IC50 = 24 nM T09572 C57IBX 25116079 IC50 = 5 nM T09572 C0WG3P 25116082 IC50 = 3 nM T09572 CV6H9C 25116306 IC50 = 747 nM T09572 CMO7K5 25116307 IC50 = 7 nM T09572 C6X3MP 25116308 IC50 = 9 nM T09572 C9FOR4 25116309 IC50 = 60 nM T09572 CV71WE 25205149 Ki = 15 nM T09572 CSY73Q 25205150 Ki = 275 nM T09572 CI60SN 25205152 Ki = 13 nM T09572 C76DEF 25205153 Ki = 24 nM T09572 CS1MG9 25205316 Ki = 25 nM T09572 CK0AS8 25205317 Ki = 11 nM T09572 C8CY6O 25205318 Ki = 5 nM T09572 CY1M9Q 25205319 Ki = 3.4 nM T09572 CP6KO3 25205320 Ki = 23 nM T09572 C86NIQ 25205321 Ki = 26 nM T09572 C8YBX7 25205493 Ki = 539 nM T09572 C0ZBD5 25205827 Ki = 19 nM T09572 CWBS82 25205829 Ki = 5.8 nM T09572 C3DF9J 25206134 Ki = 272 nM T09572 CJ94XT 25206298 Ki = 99 nM T09572 C82KIH 25206454 Ki = 2.8 nM T09572 CP7EJ2 25206612 Ki = 3.9 nM T09572 C7XQG1 25206616 Ki = 16 nM T09572 CNQ57R 25207583 Ki > 1000 nM T09572 CRCF01 30979231 IC50 = 20000 nM T09572 C8ECM1 44143489 IC50 = 375 nM T09572 C2HY7L 44143490 IC50 = 365 nM T09572 CZ08GX 44143491 IC50 > 750 nM T09572 CU54OE 44143492 IC50 = 12 nM T09572 CIN95X 44143493 IC50 = 19 nM T09572 CRJ9P8 44143494 IC50 = 24 nM T09572 CYI1M0 44143495 IC50 = 4 nM T09572 CZ81KR 44143496 IC50 = 6.7 nM T09572 CSO6G3 44143497 IC50 = 27 nM T09572 C3J2EK 44143498 IC50 = 30 nM T09572 CN7G3T 44143499 IC50 = 23 nM T09572 C12KQP 44143500 IC50 = 135 nM T09572 CKN78A 44143501 IC50 = 428 nM T09572 C2U0LK 44143502 IC50 = 41 nM T09572 CS5K8F 44143503 IC50 = 3.1 nM T09572 C21VSY 44143504 IC50 = 8.8 nM T09572 C3BUH1 44143505 IC50 = 900 nM T09572 CMY45F 44188279 Ki = 0.18 nM T09572 CT48EW 44193451 IC50 = 41 nM T09572 CV5Y8E 44193624 IC50 = 28 nM T09572 CLXI76 44193625 IC50 = 22 nM T09572 CEWK48 44193792 Ki = 4.2 nM T09572 CUT6B9 44194383 Ki = 15 nM T09572 CW29OF 44194482 Ki = 168 nM T09572 C3WE8T 44194579 Ki = 7 nM T09572 CJQ9T7 44194749 Ki = 3.6 nM T09572 C5L6WO 44194849 Ki = 4.5 nM T09572 CXM7T5 44194850 Ki = 2.7 nM T09572 C1HJE6 44194853 Ki = 6.7 nM T09572 CG65PL 44194954 Ki = 4.2 nM T09572 C76ONX 44219756 IC50 = 0.09 nM T09572 C7QS6G 44250210 IC50 = 17 nM T09572 C64ASH 44250211 IC50 = 65 nM T09572 CPG1J4 44388058 Ki = 18500 nM T09572 C7P4WR 44388077 Ki = 22500 nM T09572 C4G8DW 44388096 IC50 = 6800 nM T09572 C9RT3L 44388141 Ki = 11000 nM T09572 CR0H7L 44388201 Ki = 84 nM T09572 CL93KW 44388215 Ki = 2.2 nM T09572 C8N3YM 44388219 Ki = 13 nM T09572 C4S8VZ 44388227 Ki = 5.2 nM T09572 CFJB61 44388263 Ki = 140 nM T09572 C2CT4S 44388265 Ki = 250 nM T09572 CFQ06P 44388271 Ki = 164 nM T09572 CRIH18 44388273 Ki > 10000 nM T09572 C0E8ON 44388277 Ki = 110 nM T09572 C3GEC4 44388280 Ki > 10000 nM T09572 CEQ6Y2 44388289 Ki = 13 nM T09572 C3HEM4 44388293 Ki = 12 nM T09572 CV70XA 44388294 Ki = 14 nM T09572 CSB35R 44388303 Ki = 16 nM T09572 CR1UM2 44388308 Ki > 10000 nM T09572 CT9V3N 44388309 Ki = 4300 nM T09572 CNA6Q3 44388311 Ki = 43 nM T09572 C3OUS8 44388314 Ki = 52 nM T09572 CI3O4R 44388345 Ki > 10000 nM T09572 CQWD51 44388355 Ki = 2400 nM T09572 CU6NJ1 44388365 Ki = 34 nM T09572 C4IF0M 44388368 Ki > 10000 nM T09572 CMV89X 44388380 Ki > 10000 nM T09572 C0I5RS 44388395 Ki > 10000 nM T09572 C8W2XV 44388409 Ki = 3.1 nM T09572 CNL7F3 44388417 Ki = 5.9 nM T09572 C52KHP 44388425 Ki = 31 nM T09572 CZH08E 44388427 Ki = 130 nM T09572 CI72GN 44388428 Ki = 5.5 nM T09572 CR51FP 44388442 Ki = 8.6 nM T09572 C51CXM 44388451 Ki = 3000 nM T09572 CT0F4Y 44388559 IC50 = 299 nM T09572 CLJ51W 44389354 Ki = 48 nM T09572 CY4H3V 44389375 Ki = 64 nM T09572 C9K6JZ 44389378 Ki = 67 nM T09572 C2FA9Y 44389379 Ki = 5.3 nM T09572 CDX17Y 44389390 Ki = 96 nM T09572 CTZ7M3 44389391 Ki = 7.3 nM T09572 CDW69Y 44389392 Ki = 20 nM T09572 CE8PA6 44389403 Ki = 18 nM T09572 C6UQ3V 44389404 Ki = 14 nM T09572 CKB9H8 44389405 Ki = 82 nM T09572 C92DLV 44389406 Ki = 31 nM T09572 C07KJE 44389422 Ki = 75 nM T09572 C0COV7 44389440 Ki = 83 nM T09572 CU2PK6 44389461 Ki = 1019 nM T09572 C7ME0A 44389484 Ki = 142 nM T09572 CVZ1J6 44389490 Ki = 22 nM T09572 C6ORK9 44389509 Ki = 57 nM T09572 CT58NE 44389521 Ki = 1043 nM T09572 C51XMO 44389526 Ki = 64 nM T09572 CH1SO4 44389533 Ki = 1096 nM T09572 CX2BO7 44389546 Ki = 456 nM T09572 CA6P7D 44389590 Ki = 98 nM T09572 CTMI35 44389604 Ki = 460 nM T09572 CE25YT 44390369 IC50 = 5800 nM T09572 CFH3C2 44390385 IC50 = 960 nM T09572 C6LJC2 44390456 IC50 = 5600 nM T09572 CHGY52 44390499 IC50 = 1500 nM T09572 CK7G4S 44390706 IC50 = 5.9 nM T09572 C69OXU 44390707 IC50 = 170 nM T09572 CS16BQ 44390710 IC50 = 15 nM T09572 C9GTA2 44390713 IC50 = 9.5 nM T09572 C0B5MU 44390715 IC50 = 5 nM T09572 CBA36Y 44390726 IC50 = 2 nM T09572 C9GTB7 44390730 IC50 = 10 nM T09572 CPQ63J 44390733 IC50 = 35 nM T09572 CHO04I 44390742 IC50 = 9.4 nM T09572 CHL23R 44390748 IC50 = 1200 nM T09572 CZN1R2 44390750 IC50 = 4.5 nM T09572 C3TEB2 44390752 IC50 = 320 nM T09572 C85MAY 44390768 IC50 = 6.8 nM T09572 C5BA0Y 44390778 IC50 = 4.6 nM T09572 CN3U4V 44390787 IC50 = 38 nM T09572 CT8D4X 44393379 IC50 = 124 nM T09572 CVS4K0 44394569 IC50 = 290 nM T09572 C9GI5M 44394572 IC50 = 80 nM T09572 CAN86X 44394573 IC50 = 50 nM T09572 CSK4Z8 44394587 IC50 = 660 nM T09572 C9RD7J 44394591 IC50 = 10 nM T09572 C8HU9L 44394592 IC50 = 90 nM T09572 C79UNY 44394596 IC50 = 730 nM T09572 C63GOP 44394602 IC50 > 2000 nM T09572 CQ1M6N 44394604 IC50 = 2170 nM T09572 C24HUY 44394605 IC50 = 360 nM T09572 C9GY1S 44394606 IC50 = 30 nM T09572 C6SGC9 44394607 IC50 = 530 nM T09572 CSF04I 44394609 IC50 = 1 nM T09572 CA1H6D 44394611 IC50 = 5 nM T09572 C9Q1WO 44394628 IC50 > 2000 nM T09572 C67EUA 44394638 IC50 = 520 nM T09572 CC6HG0 44394639 IC50 = 70 nM T09572 CPK8S4 44394643 IC50 > 2000 nM T09572 CLRE30 44394644 IC50 = 340 nM T09572 C0XFU6 44394650 IC50 = 1 nM T09572 CJ78KQ 44394676 IC50 = 10 nM T09572 CY3ZO1 44394683 IC50 = 10 nM T09572 CHL3U0 44394684 IC50 = 580 nM T09572 CZ0B4R 44394697 IC50 > 10000 nM T09572 CFXI09 44394698 IC50 = 7 nM T09572 CW8RI7 44394705 IC50 = 38.6 nM T09572 CV7M6B 44394715 IC50 > 2000 nM T09572 CQ8IE0 44394725 IC50 = 7 nM T09572 CNHG32 44394726 IC50 = 2 nM T09572 CGFO71 44394763 IC50 = 10 nM T09572 CICX23 44394764 IC50 = 140 nM T09572 C57FPS 44394769 IC50 = 1.2 nM T09572 C19TJC 44394770 IC50 = 2.7 nM T09572 CJTQ96 44394774 IC50 = 306 nM T09572 C4HGJ3 44394780 IC50 > 10000 nM T09572 C1M2VQ 44394791 IC50 > 2000 nM T09572 C25PUB 44394792 IC50 = 6 nM T09572 C1NH3W 44394793 IC50 > 2000 nM T09572 CT9R3J 44394798 IC50 = 2.2 nM T09572 CLPC86 44394799 IC50 = 20.5 nM T09572 C0AQ9Y 44394800 IC50 = 1 nM T09572 C0P3SE 44394807 IC50 = 210 nM T09572 CBH9C8 44394824 IC50 = 5 nM T09572 CZN6A8 44394825 IC50 = 149 nM T09572 C6X8ZK 44394826 IC50 = 41 nM T09572 CP39MA 44394854 IC50 = 1640 nM T09572 CQ6CE2 44394855 IC50 = 240 nM T09572 C1SGN4 44394856 IC50 = 5 nM T09572 C0L8SO 44394858 IC50 > 2000 nM T09572 C35PHE 44394859 IC50 = 50 nM T09572 C6FVP1 44394860 IC50 = 30 nM T09572 CX1ZS5 44394861 IC50 = 13000 nM T09572 CHC4X1 44394863 IC50 > 2000 nM T09572 CM8P9R 44394864 IC50 = 25.6 nM T09572 CMKO91 44394866 IC50 = 10 nM T09572 C4BXR3 44394877 IC50 > 2000 nM T09572 CMR24H 44394881 IC50 > 2000 nM T09572 CYS57R 44394882 IC50 > 2000 nM T09572 CBUM52 44394883 IC50 = 80 nM T09572 COQ63G 44394890 IC50 = 100 nM T09572 CX5F2L 44394891 IC50 = 2 nM T09572 C3OVG9 44394906 IC50 > 2000 nM T09572 CTE35F 44394907 IC50 = 5.3 nM T09572 CG34PA 44394908 IC50 = 540 nM T09572 C1RD0C 44394909 IC50 = 110 nM T09572 C9I6AV 44394910 IC50 = 4700 nM T09572 C0KLA9 44394921 IC50 = 640 nM T09572 CI7RP8 44394922 IC50 = 30 nM T09572 CQ2Z0P 44394925 IC50 = 3200 nM T09572 C8G5RJ 44394926 IC50 = 960 nM T09572 C8O1VN 44394931 IC50 = 7900 nM T09572 C69ZSF 44394939 IC50 = 370 nM T09572 C90YMX 44394943 IC50 > 10000 nM T09572 CW3NK2 44394944 IC50 = 5900 nM T09572 CAOI08 44394946 IC50 = 130 nM T09572 C30MBJ 44394948 IC50 = 200 nM T09572 CTE91Q 44394958 IC50 = 1970 nM T09572 C2KM0Q 44394959 IC50 = 20 nM T09572 CB8NG3 44394961 IC50 = 640 nM T09572 C9R8NZ 44394966 IC50 = 11000 nM T09572 C49NZX 44394972 IC50 = 2500 nM T09572 CBN80V 44394973 IC50 = 2450 nM T09572 C0R9QC 44394977 IC50 > 100000 nM T09572 C8JO6R 44394978 IC50 > 100000 nM T09572 CE7HN6 44394983 IC50 = 1480 nM T09572 C1SQA9 44394986 IC50 = 250 nM T09572 C5I0CR 44394987 IC50 = 18000 nM T09572 CO5X7L 44394997 IC50 = 3500 nM T09572 CNW8A9 44394998 IC50 = 710 nM T09572 C7NM0Q 44394999 IC50 = 1920 nM T09572 C3MB6U 44395000 IC50 > 100000 nM T09572 C1JR7F 44395001 IC50 = 5800 nM T09572 C8Z5WY 44395007 IC50 = 1900 nM T09572 CY45BV 44395008 IC50 > 100000 nM T09572 CZ6G8X 44395012 IC50 = 15800 nM T09572 CKXF13 44395013 IC50 > 100000 nM T09572 CSUM01 44395019 IC50 = 140 nM T09572 CEC3Z2 44395021 IC50 = 3900 nM T09572 CGY19E 44395022 IC50 = 4800 nM T09572 CUQ04R 44395076 IC50 = 5820 nM T09572 CC48AI 44395082 IC50 = 8800 nM T09572 C67MQP 44396196 IC50 = 8200 nM T09572 CDH9A0 44396800 Ki = 3 nM T09572 C1Q3KE 44396807 Ki = 2 nM T09572 CK24UL 44396904 Ki = 310 nM T09572 C06GEV 44396952 IC50 = 90 nM T09572 C34UGT 44396975 Ki = 63 nM T09572 C3QE2M 44396985 Ki = 61 nM T09572 CJO81G 44397008 IC50 = 50 nM T09572 C5LY2S 44397009 IC50 = 110 nM T09572 CG9L7A 44397018 Ki = 3 nM T09572 CCO72P 44397026 IC50 = 50 nM T09572 C4V9XD 44397031 Ki = 10 nM T09572 C1YAO3 44397033 IC50 = 4300 nM T09572 CR7I9Z 44397048 IC50 = 230 nM T09572 C6DTI3 44397052 IC50 > 2000 nM T09572 CXP1H2 44397086 Ki = 3 nM T09572 CZXN03 44397087 Ki = 7 nM T09572 CQZ9M6 44397095 Ki = 3 nM T09572 C5NR9X 44397099 IC50 = 5190 nM T09572 CSY42I 44397103 Ki = 6000 nM T09572 C0DE8P 44397114 Ki = 1 nM T09572 C8VPO7 44397120 IC50 = 510 nM T09572 CJ3HW9 44397126 Ki = 190 nM T09572 C1O0AT 44397127 IC50 = 50 nM T09572 CVD8J2 44397128 IC50 = 60 nM T09572 CN26GO 44397145 Ki = 1800 nM T09572 C2I9VT 44397163 Ki = 37 nM T09572 CD15XJ 44397167 Ki = 19 nM T09572 C41YAD 44397168 Ki = 3300 nM T09572 CT3IG2 44397174 IC50 > 10000 nM T09572 C0IOB2 44397175 IC50 = 300 nM T09572 CM83JY 44397194 IC50 = 20 nM T09572 CO8EI5 44397200 Ki = 320 nM T09572 CFY3U9 44397202 IC50 = 10 nM T09572 CR6YG0 44397203 Ki > 10000 nM T09572 C1MQ3T 44397215 IC50 = 320 nM T09572 CQ73UR 44397221 IC50 = 90 nM T09572 CL8IY3 44397227 Ki = 900 nM T09572 C4CQT2 44397243 Ki = 3400 nM T09572 C58DRB 44397245 Ki = 4 nM T09572 CZ30KL 44397254 Ki = 3 nM T09572 C92RCK 44397262 IC50 = 30 nM T09572 CB2ZN8 44397263 IC50 > 2000 nM T09572 C5IXH8 44397273 Ki = 5 nM T09572 CSI3G7 44397278 IC50 = 490 nM T09572 CX3ED1 44397288 Ki = 2 nM T09572 C6DZQ0 44397293 Ki = 4 nM T09572 CFP9Y1 44397302 Ki = 14 nM T09572 CZK80P 44397303 IC50 = 1040 nM T09572 CZKY29 44397309 Ki = 12 nM T09572 C7R3EV 44397310 IC50 = 110 nM T09572 C9IZO5 44397312 Ki = 2400 nM T09572 CLC7N8 44397323 Ki = 150 nM T09572 CP6I4E 44397329 IC50 = 1950 nM T09572 CB5ZQ7 44397330 IC50 > 2000 nM T09572 C9X3JV 44397350 Ki = 16 nM T09572 CV72OU 44397425 IC50 = 90 nM T09572 C82FLB 44397454 IC50 = 2990 nM T09572 CMJ67E 44397476 IC50 = 3 nM T09572 C9AM8F 44397477 IC50 > 2000 nM T09572 CSRG09 44397479 Ki = 2 nM T09572 CI2VP7 44397480 IC50 = 320 nM T09572 C6LJB5 44397497 Ki = 5 nM T09572 CS07BY 44397560 IC50 = 120 nM T09572 CR2DJ8 44397605 IC50 = 1610 nM T09572 C5B2YW 44397606 IC50 = 280 nM T09572 CPB7Q4 44397630 Ki = 2 nM T09572 CS4IW6 44397636 IC50 = 330 nM T09572 C0QM4W 44397716 IC50 = 1560 nM T09572 C4HR6C 44399507 Ki = 7.1 nM T09572 CH39TA 44399610 Ki = 2.7 nM T09572 CL06NB 44401276 IC50 > 10000 nM T09572 CDS4Y1 44401368 IC50 = 6700 nM T09572 C93HAW 44401395 IC50 = 2700 nM T09572 C4RN8A 44401449 IC50 = 83 nM T09572 C49USD 44401460 IC50 > 10000 nM T09572 CHGX51 44401508 IC50 = 2900 nM T09572 CIKD90 44401552 IC50 = 2900 nM T09572 C8VQ3B 44401591 IC50 = 1900 nM T09572 CT46VH 44401616 IC50 = 810 nM T09572 CIXE76 44401626 IC50 = 140 nM T09572 CER15G 44401671 IC50 = 6000 nM T09572 CR1D2K 44402861 Ki > 100000 nM T09572 CW4Z1L 44403445 IC50 = 370 nM T09572 C4UDG8 44403454 IC50 = 370 nM T09572 CT6IX9 44403467 IC50 = 6 nM T09572 CBN6J3 44403468 IC50 = 20 nM T09572 CRWC57 44403471 IC50 = 110 nM T09572 CT0U6C 44403472 IC50 = 80 nM T09572 C5Q0OF 44403473 IC50 = 2010 nM T09572 CJ1U2V 44403474 IC50 = 30 nM T09572 C3Y2ST 44403477 IC50 = 9 nM T09572 CHZI37 44403478 IC50 = 680 nM T09572 C1JRE0 44403479 IC50 = 70 nM T09572 CF6QJ8 44403480 IC50 = 30 nM T09572 C1FOP8 44403483 IC50 = 560 nM T09572 CT2GD3 44403484 IC50 = 260 nM T09572 C1P5JF 44403486 IC50 = 1980 nM T09572 CF7Z6C 44403487 IC50 = 20 nM T09572 CE27XC 44403490 IC50 = 160 nM T09572 CI4S5Z 44403491 IC50 = 220 nM T09572 C5I7ZO 44403492 IC50 = 160 nM T09572 CUZH85 44403493 IC50 = 20 nM T09572 CWCJ58 44403498 IC50 = 90 nM T09572 C6OWP7 44403499 IC50 = 50 nM T09572 CE9W5D 44403500 IC50 = 410 nM T09572 CSP0T1 44403501 IC50 = 60 nM T09572 CXH8U1 44403505 IC50 = 40 nM T09572 CLK27J 44403506 IC50 = 30 nM T09572 C5D1NZ 44403507 IC50 = 20 nM T09572 CWP5R7 44403511 IC50 = 9 nM T09572 C39ZVY 44403513 IC50 = 9 nM T09572 CHS0Y9 44403516 IC50 = 70 nM T09572 C1V6BP 44403517 IC50 = 4 nM T09572 CEJF46 44403518 IC50 = 6 nM T09572 C5UG0H 44403522 IC50 = 20 nM T09572 C8I1JU 44403523 IC50 = 10 nM T09572 C41YLX 44403524 IC50 = 60 nM T09572 CNW95X 44403527 IC50 = 90 nM T09572 CFS35E 44403528 IC50 = 50 nM T09572 CB02DH 44403533 IC50 = 390 nM T09572 C65YJN 44403535 IC50 = 190 nM T09572 C4U3FN 44403538 IC50 = 70 nM T09572 C19IBE 44403539 IC50 = 140 nM T09572 C2OMY6 44403547 IC50 = 410 nM T09572 C0TO1J 44403548 IC50 = 10 nM T09572 CQ08CG 44403733 IC50 = 1800 nM T09572 CZE89R 44403747 IC50 = 95 nM T09572 CR7BQ9 44403748 IC50 = 438 nM T09572 CQ4W5H 44403749 IC50 = 442 nM T09572 C81ISR 44403750 IC50 = 224 nM T09572 CLGA83 44403765 IC50 = 6.1 nM T09572 CBA93S 44403849 IC50 > 10000 nM T09572 CD3FE4 44405399 Ki = 287 nM T09572 CQDZ37 44405408 IC50 = 50 nM T09572 C2DAJ8 44405409 IC50 = 330 nM T09572 CA75TW 44405412 IC50 = 5200 nM T09572 C8A2RI 44405415 IC50 = 30 nM T09572 CW5KU8 44405417 Ki = 159 nM T09572 CVP74K 44405418 Ki = 48 nM T09572 C0N4IL 44405421 Ki = 48 nM T09572 C5F2LI 44405430 IC50 = 4500 nM T09572 C5T9CU 44405431 IC50 = 1380 nM T09572 C79OPX 44405435 Ki = 23 nM T09572 CDJF17 44405436 Ki = 70 nM T09572 CT42XM 44405437 Ki = 151 nM T09572 CF57KL 44405439 Ki = 18 nM T09572 C37XOM 44405444 Ki = 76 nM T09572 C74WZI 44405458 IC50 > 2000 nM T09572 C5V3EU 44405459 IC50 = 200 nM T09572 CW80JL 44405461 Ki = 16 nM T09572 CBS4P2 44405463 IC50 = 50 nM T09572 C5KLO6 44405464 IC50 = 5 nM T09572 CJRW91 44405468 IC50 = 40 nM T09572 C29JXR 44405477 IC50 = 850 nM T09572 C27IXA 44405481 IC50 = 1060 nM T09572 CB78MN 44405482 IC50 = 70 nM T09572 C9V7MC 44405486 IC50 = 520 nM T09572 CX64ET 44405487 IC50 = 220 nM T09572 C16CPT 44405488 IC50 = 280 nM T09572 CN4KP9 44405501 Ki = 31 nM T09572 C1T3AR 44405517 IC50 = 440 nM T09572 CTW14K 44405518 IC50 = 1820 nM T09572 CC38GX 44405519 IC50 = 70 nM T09572 CJ2OV1 44405557 IC50 = 930 nM T09572 CH7XF0 44405560 IC50 = 20 nM T09572 C1GA2K 44405570 IC50 = 50 nM T09572 CN2W1H 44405612 IC50 = 20 nM T09572 CB79VL 44405618 IC50 = 20 nM T09572 CTI27L 44405619 IC50 = 560 nM T09572 CU08QO 44405645 IC50 = 40 nM T09572 C3H4OS 44405646 IC50 = 20 nM T09572 CD4H0S 44405651 IC50 = 9 nM T09572 C7DY8R 44407478 IC50 > 10000 nM T09572 C7TXS3 44407479 IC50 = 2540 nM T09572 CY70WO 44407629 IC50 = 2 nM T09572 C29UTK 44407667 IC50 = 17 nM T09572 CBL19U 44407710 IC50 = 3.7 nM T09572 CBU72F 44407711 IC50 = 83 nM T09572 C0BY6Z 44407836 IC50 = 4.7 nM T09572 CP5D3Y 44407860 IC50 = 91 nM T09572 C3JLT1 44407870 IC50 = 14 nM T09572 C8TP0Q 44407875 IC50 = 3.7 nM T09572 C8FTO7 44407934 IC50 = 2100 nM T09572 C7MEY5 44407944 IC50 = 33 nM T09572 CRS49X 44407950 IC50 = 2760 nM T09572 CB0LM3 44407951 IC50 = 125 nM T09572 CUEI62 44407956 IC50 = 44 nM T09572 CU34HG 44407965 IC50 > 10000 nM T09572 CV9R8K 44407966 IC50 = 105 nM T09572 CYOP29 44407967 IC50 = 474 nM T09572 CK13PD 44407989 IC50 = 6970 nM T09572 CF3X7M 44407990 IC50 > 10000 nM T09572 CR8B7D 44407991 IC50 = 5.7 nM T09572 CWUS42 44407997 IC50 = 9460 nM T09572 C70DWK 44408013 IC50 = 23 nM T09572 CG9HB0 44408014 IC50 = 3280 nM T09572 CA72TP 44408020 IC50 = 568 nM T09572 C6IT1B 44408027 IC50 = 15 nM T09572 CVS92Y 44408028 IC50 = 7.1 nM T09572 CP8A0C 44408081 IC50 = 210 nM T09572 CG5JN8 44408093 IC50 = 162 nM T09572 CT9Q7Z 44408099 IC50 = 271 nM T09572 CU4JK5 44408108 IC50 = 5.3 nM T09572 COGK24 44408109 IC50 = 2.4 nM T09572 CBJY53 44408117 IC50 = 18 nM T09572 CUS7R1 44409479 Ki = 15 nM T09572 C1DTI6 44409527 Ki = 15.1 nM T09572 CKEP27 44409689 Ki = 974 nM T09572 CYP37K 44410821 IC50 = 5 nM T09572 CJI8T3 44410823 IC50 = 62 nM T09572 C01JXU 44410838 IC50 = 72 nM T09572 C1LYC9 44410849 IC50 = 0.9 nM T09572 CGF17I 44410876 IC50 = 12 nM T09572 CF0O7N 44410878 IC50 = 34 nM T09572 CL1XV7 44410904 IC50 = 53 nM T09572 C4P5TW 44410944 IC50 = 12 nM T09572 CFSD50 44412624 Ki = 51 nM T09572 C1CPT2 44412682 Ki = 46 nM T09572 CG6J5R 44412683 Ki = 92 nM T09572 CQ7P1N 44412686 Ki = 48 nM T09572 CVJF97 44412837 Ki = 26 nM T09572 CRPQ04 44412852 Ki = 1.2 nM T09572 CV1ZX4 44412960 Ki = 193 nM T09572 C43CDI 44413138 Ki = 132 nM T09572 C2SOJ1 44413259 Ki = 95 nM T09572 C8OT1W 44413271 Ki = 77 nM T09572 C1AJ8V 44413283 Ki = 3.9 nM T09572 CHG2A7 44413297 Ki = 10.3 nM T09572 C6V5YR 44413299 Ki = 31 nM T09572 C7PC5N 44413309 Ki = 26 nM T09572 C4YMR8 44413312 Ki = 31 nM T09572 CXC97Y 44413326 IC50 = 130 nM T09572 C0IBW4 44413345 Ki = 464 nM T09572 C9U8FY 44413382 Ki = 7.2 nM T09572 CDG5Q2 44413398 Ki = 99 nM T09572 C64UZT 44413428 Ki = 174 nM T09572 CK8C1H 44413470 Ki = 15.5 nM T09572 C34LQB 44413471 Ki = 45 nM T09572 CG7KI9 44413472 Ki = 20 nM T09572 CGY94E 44413473 Ki = 10.1 nM T09572 C7X5HF 44413474 Ki = 10.3 nM T09572 CCKU08 44413475 Ki = 15 nM T09572 CS5WN4 44413480 Ki = 64 nM T09572 CB5GI6 44414309 Ki = 3 nM T09572 C3IB1L 44414310 Ki = 8.8 nM T09572 C79XQN 44414318 Ki = 4.4 nM T09572 CJ1V0F 44414319 Ki = 13 nM T09572 C9MV4A 44414327 Ki = 10 nM T09572 CZI1Y9 44414342 Ki = 24 nM T09572 CS5VO0 44414356 Ki = 24 nM T09572 C2XK7V 44414357 Ki = 14 nM T09572 C5M6ZU 44414368 Ki = 120 nM T09572 CIJ8D5 44414375 Ki = 4.8 nM T09572 C52EQN 44414391 Ki = 7.2 nM T09572 CMV9H6 44414392 Ki = 13 nM T09572 C2N7PZ 44414399 Ki = 3.1 nM T09572 CE36JR 44414432 Ki = 4.1 nM T09572 C2BXH0 44414444 Ki = 25 nM T09572 C1X5TM 44414451 Ki = 2 nM T09572 CXQK29 44414455 Ki = 18 nM T09572 C3CA5G 44414461 Ki = 57 nM T09572 CU8VR5 44414464 Ki = 15.1 nM T09572 C2D9BH 44414465 Ki = 115 nM T09572 CEL21T 44414466 Ki = 28 nM T09572 CKB82R 44414475 Ki = 2.1 nM T09572 CB5F4W 44414481 Ki = 29 nM T09572 CY1VH7 44414483 Ki = 28 nM T09572 C96BYD 44414497 Ki = 1.6 nM T09572 C3DP8X 44414499 Ki = 19 nM T09572 CHG0S9 44414506 Ki = 56 nM T09572 CH7P4X 44414518 Ki = 10 nM T09572 CG7J0K 44414520 Ki = 1.4 nM T09572 CTE9S2 44414522 Ki = 138 nM T09572 CX2F6A 44414528 Ki = 8.6 nM T09572 CJ0FN4 44414540 Ki = 7.1 nM T09572 CL0H1X 44414542 Ki = 78 nM T09572 CR1CS5 44414552 Ki = 43 nM T09572 CBJF79 44414570 Ki = 16 nM T09572 C7E6RX 44414571 Ki = 4.7 nM T09572 C2I9CV 44414576 Ki = 5.4 nM T09572 CSEN81 44414589 Ki = 5.4 nM T09572 C97FHL 44414600 Ki = 2.6 nM T09572 C10IPW 44414601 Ki = 46 nM T09572 CS1B0T 44414606 Ki = 15 nM T09572 CG6R9J 44414622 Ki = 2.7 nM T09572 C6E7RW 44414649 Ki = 8.5 nM T09572 C9KHE1 44414650 Ki = 17 nM T09572 C40PGW 44414651 Ki = 139 nM T09572 CWIM26 44414654 Ki = 6.8 nM T09572 CGI4F7 44415364 Ki = 10.47 nM T09572 CPJ4V5 44415378 Ki = 18.62 nM T09572 CWJE81 44415381 Ki = 630 nM T09572 CC25QM 44415385 Ki = 4786.3 nM T09572 CMV57G 44415389 Ki = 13 nM T09572 CN1M4Z 44415396 Ki = 398.11 nM T09572 CRHQ87 44415401 Ki = 39.81 nM T09572 C29JXK 44415402 Ki = 23.99 nM T09572 C1T2DR 44415407 Ki = 630.96 nM T09572 C83UJR 44415409 Ki = 51 nM T09572 CRUT01 44415410 Ki = 53 nM T09572 C75SYA 44415413 Ki = 16 nM T09572 CR34JS 44415414 Ki = 41.69 nM T09572 CH91UG 44415419 Ki = 1000 nM T09572 C9WRN5 44415425 Ki = 33.88 nM T09572 C7VT5P 44415426 Ki = 53.7 nM T09572 CV9S7J 44415427 Ki = 51 nM T09572 CFZ90J 44415431 Ki = 43.65 nM T09572 C09SEJ 44415439 Ki = 38 nM T09572 C0TZ3O 44415440 Ki = 28.84 nM T09572 CPM3R9 44415446 Ki = 28 nM T09572 C7NH2F 44415451 Ki = 8 nM T09572 C5IV2C 44415459 Ki = 33 nM T09572 CL1KM8 44415460 Ki = 25.7 nM T09572 CGHJ29 44415461 Ki = 14 nM T09572 COW3P7 44415462 Ki = 26.92 nM T09572 COLW46 44415463 Ki = 47.86 nM T09572 C5Z9UM 44415465 Ki > 10000 nM T09572 CU2LQ5 44415466 Ki = 3981.07 nM T09572 CX76TL 44415467 Ki = 73 nM T09572 CTS2L6 44415483 Ki = 16.6 nM T09572 CI05LE 44415491 Ki = 22 nM T09572 CQKB40 44415501 Ki = 109.65 nM T09572 CO8X2W 44415512 Ki = 180 nM T09572 CN9GY5 44415516 Ki = 48.98 nM T09572 C0OG4J 44415524 Ki = 14 nM T09572 C86OHN 44415525 Ki = 20.89 nM T09572 CL17YI 44415526 Ki = 19.95 nM T09572 CY6C2D 44415533 Ki = 18.62 nM T09572 C6HSF3 44416140 Ki = 41 nM T09572 CZG1L2 44416172 Ki = 77 nM T09572 CZ38VN 44416173 Ki = 87 nM T09572 CT79MH 44416174 Ki = 799 nM T09572 C9FT7Y 44416178 Ki = 46 nM T09572 CV8JU0 44416212 IC50 = 25.12 nM T09572 CN78HS 44416223 Ki = 95 nM T09572 CKD7I4 44416224 Ki = 191 nM T09572 CKP27D 44416225 Ki = 77 nM T09572 C58WVT 44416231 IC50 = 5.012 nM T09572 CE93MV 44416232 IC50 = 199.53 nM T09572 CAO4W7 44416255 IC50 = 1584.89 nM T09572 C5B3IQ 44416261 Ki = 24 nM T09572 CBC5O3 44416272 IC50 = 25.12 nM T09572 CITW25 44416275 Ki = 927 nM T09572 C2AO6C 44416287 Ki = 718 nM T09572 C9F2PM 44416296 IC50 = 19.95 nM T09572 C0LQ3D 44416297 IC50 = 1258.93 nM T09572 CVXO51 44416302 IC50 = 5.012 nM T09572 CD9J7M 44416303 IC50 = 3162.28 nM T09572 CGC7V2 44416310 Ki = 108 nM T09572 C8IPQ2 44416311 Ki = 73 nM T09572 CUN0J8 44416314 IC50 = 1.259 nM T09572 CKJ1N7 44416315 IC50 = 6.31 nM T09572 CFI41O 44416316 IC50 = 1.585 nM T09572 CN4O2X 44416322 Ki = 43 nM T09572 CHL8D7 44416336 IC50 = 1 nM T09572 CB7H1J 44416337 IC50 = 2.512 nM T09572 CV13DW 44416344 Ki > 1000 nM T09572 C8XCL1 44416346 Ki = 455 nM T09572 C5SI3O 44416348 IC50 = 12.59 nM T09572 CRJ97I 44416350 IC50 = 100 nM T09572 CPUD71 44416357 Ki = 115 nM T09572 CLXG42 44416362 IC50 = 3981.07 nM T09572 CF19EV 44416363 IC50 = 125.89 nM T09572 CU64KI 44416364 Ki = 35 nM T09572 CX59PC 44416376 IC50 = 6.31 nM T09572 CA98PR 44416377 IC50 = 3.162 nM T09572 CQV5J1 44416381 Ki = 168 nM T09572 C4BJR5 44416388 Ki = 25.12 nM T09572 CB7P8K 44416389 Ki = 158.49 nM T09572 CP7H2Q 44416390 Ki = 5.012 nM T09572 CF0BM8 44416391 Ki = 414 nM T09572 CRO95N 44416402 Ki = 398.11 nM T09572 CFUA54 44416405 Ki = 4.9 nM T09572 CAE2D0 44416428 Ki = 251.19 nM T09572 C8P2XM 44416451 Ki < 6309.57 nM T09572 C32IYJ 44416472 Ki = 251.19 nM T09572 C2F3EY 44416474 Ki = 102 nM T09572 C70GBX 44416475 Ki = 1408 nM T09572 CNL35D 44416479 Ki = 31.62 nM T09572 CVF1B8 44416480 Ki = 251.19 nM T09572 C4AOQ9 44416495 Ki = 79.43 nM T09572 C4SP0A 44416498 Ki = 39.81 nM T09572 C42WEU 44416502 Ki = 50.12 nM T09572 C7IB2N 44416503 Ki = 50.12 nM T09572 CVA3M1 44416504 Ki < 10000 nM T09572 C15TAE 44416521 Ki = 39.81 nM T09572 CO0QD7 44416522 Ki = 2511.89 nM T09572 CEH6A9 44416536 Ki < 10000 nM T09572 C4L8UP 44416539 Ki = 39.81 nM T09572 C79YPB 44416540 Ki < 10000 nM T09572 CPE1L9 44416553 Ki = 50.12 nM T09572 C3UIT1 44416554 Ki = 79.43 nM T09572 CF0E9H 44416559 Ki = 125.89 nM T09572 C1VT2K 44416561 Ki = 63.1 nM T09572 CBP2N5 44416579 Ki = 199.53 nM T09572 C75GYI 44416580 Ki = 501.19 nM T09572 CJ4D5N 44416584 Ki = 79.43 nM T09572 C9CD8Z 44416585 Ki = 158.49 nM T09572 C6H0BL 44416586 Ki = 25.12 nM T09572 C9VS6Z 44416587 Ki = 1153 nM T09572 C87FGN 44416606 Ki = 50.12 nM T09572 CAF18G 44416607 Ki = 60 nM T09572 CC1Y0W 44416623 Ki = 5011.87 nM T09572 CZ7W0E 44416624 Ki < 10000 nM T09572 C4RS6H 44416627 Ki = 310 nM T09572 CF3HG1 44416628 Ki = 3544 nM T09572 C8A5HU 44416629 Ki = 31 nM T09572 CT4DU9 44416650 Ki = 20119 nM T09572 C7JV9E 44416651 Ki = 0.631 nM T09572 CFZ0H1 44416664 Ki = 63.1 nM T09572 CN3UQ7 44416670 Ki = 1.995 nM T09572 C8ZI4H 44416671 Ki = 0.9 nM T09572 CGB3S0 44416689 Ki = 803 nM T09572 C6BD0R 44416711 Ki = 199.53 nM T09572 CE5MY9 44416713 Ki = 195 nM T09572 CSRK76 44416714 Ki = 19.95 nM T09572 C1YV3D 44416735 Ki = 79.43 nM T09572 CV7BA5 44416736 Ki < 10000 nM T09572 C0V4BK 44416737 Ki = 142 nM T09572 C95RCN 44416738 Ki = 310 nM T09572 CX0R4H 44416751 IC50 = 100 nM T09572 CJ08ZR 44416753 Ki = 25 nM T09572 C3O7GK 44416757 Ki = 3.981 nM T09572 CA28XT 44416777 IC50 = 5.012 nM T09572 C16WUL 44416781 Ki = 3600 nM T09572 CY6T2S 44416782 Ki = 18 nM T09572 C0SX4T 44416786 Ki = 12.59 nM T09572 CK1UJ6 44416797 Ki = 1000 nM T09572 CD2U4N 44416798 Ki = 316.23 nM T09572 C9R1UT 44416800 Ki = 1.585 nM T09572 CMHX86 44416801 Ki = 5 nM T09572 CGMX09 44416814 IC50 = 6.31 nM T09572 CL53YH 44416815 IC50 = 6.31 nM T09572 CAT0B7 44416816 Ki = 2511.89 nM T09572 C4OX7Y 44416817 Ki = 1995.26 nM T09572 CSRH79 44416828 IC50 = 25.12 nM T09572 C0VJ9B 44416833 Ki = 133 nM T09572 C94QFT 44416837 IC50 = 1.995 nM T09572 CAZW24 44416838 IC50 = 5.012 nM T09572 CD9Q0Y 44416839 Ki = 136 nM T09572 C81JPB 44416840 Ki = 110 nM T09572 CRMS24 44416841 Ki = 794.33 nM T09572 C0WCI8 44416845 IC50 = 6.31 nM T09572 C7SIK0 44416851 IC50 = 31.62 nM T09572 CP64OW 44416857 IC50 = 1.585 nM T09572 C1UMD2 44416858 IC50 = 31.62 nM T09572 C4W8ST 44416859 Ki = 1.9 nM T09572 CG46MT 44416862 Ki = 6 nM T09572 CKNF68 44416871 IC50 = 19.95 nM T09572 CI35XF 44416872 IC50 = 5.012 nM T09572 CP4YB0 44416875 IC50 = 3.981 nM T09572 CT62LG 44416877 Ki = 2.4 nM T09572 C8ELH9 44416880 Ki = 500 nM T09572 C76SRF 44416881 Ki = 2 nM T09572 CWS2B9 44416890 IC50 = 3.162 nM T09572 CDNH81 44416895 Ki = 3.7 nM T09572 C2FX5H 44416898 Ki = 10 nM T09572 CPNY68 44416910 Ki = 197 nM T09572 CLP16U 44416911 Ki = 1.585 nM T09572 C0X5HE 44416916 Ki = 63.1 nM T09572 C0OMX6 44416923 IC50 > 1000 nM T09572 CE0SK3 44416928 Ki = 126 nM T09572 CB9RO3 44416929 Ki = 91 nM T09572 CZ8CS2 44416935 IC50 = 5.012 nM T09572 C5G7KA 44416946 IC50 > 1000 nM T09572 CC9KR4 44416947 IC50 > 1000 nM T09572 C74ATQ 44416949 IC50 = 25.12 nM T09572 C87RVU 44416955 IC50 = 5.012 nM T09572 C5MI0P 44416956 IC50 = 12.59 nM T09572 C5C7QR 44416964 IC50 > 1000 nM T09572 CILD84 44416966 Ki = 773 nM T09572 C5MY6P 44416968 Ki = 79.43 nM T09572 C7BI9T 44416969 Ki = 10 nM T09572 CIEB89 44416970 Ki = 10 nM T09572 C9WRP8 44416975 IC50 = 2511.89 nM T09572 CW2I3N 44416976 IC50 = 10 nM T09572 C9QU0R 44416989 Ki = 7.943 nM T09572 C8BQ3P 44416990 Ki = 31.62 nM T09572 CTC30S 44416995 IC50 = 12.59 nM T09572 C5C1PE 44417017 IC50 = 170 nM T09572 C0DV8X 44417021 IC50 = 2.512 nM T09572 CGNK93 44417022 IC50 = 7.943 nM T09572 C05LZR 44417024 Ki = 2.512 nM T09572 CZ5SQ3 44417025 Ki = 5 nM T09572 CFPC71 44417043 IC50 = 15.85 nM T09572 CZ4Q5J 44417044 IC50 = 3.162 nM T09572 C2LW3E 44417061 Ki = 84 nM T09572 CE8KJ6 44417066 IC50 = 5.012 nM T09572 C0NI5V 44417067 IC50 = 15.85 nM T09572 C0A2FS 44417069 Ki = 15.85 nM T09572 CK92GD 44417083 IC50 = 7.943 nM T09572 CCX9R4 44417140 IC50 = 31.62 nM T09572 CXLI76 44417145 IC50 = 6.31 nM T09572 CQP8L9 44417146 IC50 = 5.012 nM T09572 C7WY1L 44417150 IC50 = 10 nM T09572 C0YZ7M 44417151 IC50 = 6.31 nM T09572 CT3KX7 44417481 IC50 > 2000 nM T09572 C0V7EJ 44417821 EC50 = 370 nM T09572 CA61IW 44417822 IC50 = 10000 nM T09572 C0Y8UH 44417823 EC50 = 120 nM T09572 CYAD92 44417824 IC50 = 4000 nM T09572 CG0E3N 44417825 IC50 = 1700 nM T09572 CPX53N 44417827 IC50 = 1100 nM T09572 CU72ZV 44417828 Ki = 27 nM T09572 C46RHE 44417829 Ki = 56 nM T09572 C8AQU5 44417830 Ki = 1000 nM T09572 CR0G9W 44417831 Ki = 286 nM T09572 CYNX47 44417832 IC50 = 0.7 nM T09572 CC0P6Y 44417833 Ki = 133 nM T09572 CLHV60 44417834 Ki > 100000 nM T09572 CDT9M1 44417835 Ki = 8.6 nM T09572 C3F4ZC 44417836 Ki = 86 nM T09572 CAO59Y 44417837 Ki = 170 nM T09572 C0NPX2 44417838 EC50 = 500 nM T09572 C8QB4F 44417839 Ki = 36 nM T09572 C1OL9Y 44417840 Ki = 40 nM T09572 CPF38S 44417841 Ki = 18 nM T09572 C7D4FK 44417842 Ki = 9 nM T09572 C8XC5O 44417843 IC50 = 2.3 nM T09572 CC26DZ 44417844 EC50 = 71 nM T09572 CNQ02C 44417845 EC50 = 40 nM T09572 C1EHB3 44417846 IC50 = 1.4 nM T09572 C3QP7X 44417847 EC50 = 3600 nM T09572 C9TN8Y 44417848 EC50 = 740 nM T09572 CO51ID 44417849 Ki = 232 nM T09572 C96QJO 44417850 Ki = 7 nM T09572 CNX80R 44417851 Ki > 100000 nM T09572 CAI3K8 44417852 Ki = 484 nM T09572 CA7T1X 44417853 Ki = 67 nM T09572 CT7WS4 44417854 Ki = 65 nM T09572 C1MEX3 44417855 Ki = 13 nM T09572 CZO51X 44417856 EC50 = 990 nM T09572 C1JQ5P 44417857 EC50 = 310 nM T09572 CG05EA 44417858 IC50 = 190 nM T09572 CP8AF3 44417859 Ki = 32 nM T09572 CP72QS 44417860 Ki = 62 nM T09572 C1W4VB 44417861 Ki = 12 nM T09572 C05HMG 44417862 Ki = 17 nM T09572 CB10YP 44417863 Ki = 28.2 nM T09572 CB62CN 44417864 IC50 = 95 nM T09572 CQNF68 44417865 Ki = 125 nM T09572 CU7XD8 44417866 IC50 = 1100 nM T09572 C57FVT 44417867 IC50 = 130 nM T09572 CV4EF6 44417868 Ki = 441 nM T09572 CL8X5U 44417869 Ki = 25 nM T09572 C0ODM7 44417870 Ki = 625 nM T09572 C3FO0H 44417871 Ki = 23 nM T09572 CT8FJ0 44417872 Ki = 8070 nM T09572 CI60HL 44417873 EC50 = 910 nM T09572 CC61GR 44417874 IC50 = 9 nM T09572 C6A2YW 44417875 EC50 = 118 nM T09572 CCD0P3 44417876 Ki = 142 nM T09572 CGWI26 44417877 EC50 = 520 nM T09572 CT27KD 44417878 Ki = 505 nM T09572 CA34LP 44417879 Ki = 2.5 nM T09572 C42RJO 44417880 Ki = 205 nM T09572 CU9JD6 44417881 Ki = 136 nM T09572 CN25SX 44417882 Ki > 100000 nM T09572 C21ZCB 44417883 IC50 = 1797 nM T09572 C6HJ3K 44417885 Ki = 169 nM T09572 CRT85J 44417886 EC50 = 2800 nM T09572 CG1WM8 44417887 Ki = 3.3 nM T09572 C89TAB 44417888 IC50 = 20 nM T09572 CK76AM 44417889 Ki = 32 nM T09572 CPE50S 44417890 IC50 = 76 nM T09572 CQS6G2 44417891 Ki = 93 nM T09572 CO0U5H 44417892 IC50 = 300 nM T09572 CAK9U7 44417893 Ki = 52000 nM T09572 C26CUN 44417894 IC50 = 13 nM T09572 C35KLS 44417895 Ki = 146 nM T09572 CL5XO4 44417897 IC50 = 11 nM T09572 CKI1W2 44417898 IC50 = 750 nM T09572 CM9QI8 44417899 IC50 = 21 nM T09572 C6UAH2 44417900 Ki = 2480 nM T09572 CWO51Q 44417901 Ki = 145 nM T09572 CI16UJ 44417902 IC50 = 1267 nM T09572 C0US4Z 44417903 IC50 = 18 nM T09572 C8GK5Q 44417904 Ki = 24 nM T09572 CHC7G9 44417905 Ki = 11 nM T09572 C9BDI1 44417906 IC50 = 95 nM T09572 CC3S6F 44417907 IC50 = 3700 nM T09572 C3GW2E 44417908 Ki = 94000 nM T09572 CKQ92G 44417909 Ki = 22 nM T09572 CN2G7U 44417910 IC50 = 43 nM T09572 C46KMH 44417911 IC50 = 4 nM T09572 C2XJW5 44417912 Ki = 5294 nM T09572 CPDW02 44417913 Ki = 184 nM T09572 CY46AB 44417914 Ki = 270000 nM T09572 C9HN5T 44417915 IC50 = 800 nM T09572 C5HA7X 44417916 Ki = 18 nM T09572 CM2UC6 44417917 IC50 = 25 nM T09572 CD62PS 44417918 Ki = 100000 nM T09572 CW1D3V 44417919 Ki = 11 nM T09572 CCU69N 44417920 Ki = 62000 nM T09572 CFR6H4 44417921 IC50 = 12 nM T09572 C3CM4J 44417922 Ki = 12 nM T09572 CH0T1F 44417923 Ki = 15000 nM T09572 C4WU0N 44417924 Ki = 30000 nM T09572 CTUV23 44417925 IC50 = 10 nM T09572 CE96RJ 44417926 Ki = 20 nM T09572 C27PHW 44417927 Ki = 47 nM T09572 CEZH78 44417928 Ki = 103 nM T09572 CT0B1U 44417929 Ki = 8700 nM T09572 CB8IZ1 44417930 IC50 = 3 nM T09572 CPO9R1 44417931 IC50 = 622 nM T09572 C7F4LM 44417933 Ki = 2482 nM T09572 CS9AZ3 44417934 Ki = 82 nM T09572 CH08OA 44417936 IC50 = 2010 nM T09572 C7W8KZ 44417937 IC50 = 166 nM T09572 CH3QM1 44417938 IC50 = 47 nM T09572 CP1U0Z 44417939 IC50 = 19 nM T09572 C3B4LO 44417940 IC50 = 180 nM T09572 C7IJZ9 44417941 IC50 = 25 nM T09572 CP5K2A 44417942 IC50 = 2700 nM T09572 CM6H8T 44417943 IC50 = 45 nM T09572 CHSE12 44417944 EC50 = 110 nM T09572 C89EBO 44417945 IC50 = 3 nM T09572 C42OAE 44417946 IC50 = 763 nM T09572 CQ7M6F 44417947 EC50 = 250 nM T09572 C70AVF 44417948 EC50 = 68 nM T09572 CZK6C5 44417949 IC50 = 4 nM T09572 C3WT1V 44417950 Ki = 15 nM T09572 CM76IN 44417952 IC50 = 96 nM T09572 C6F9MN 44417953 Ki = 23 nM T09572 C3P1JG 44417954 Ki = 727 nM T09572 CLOU53 44417955 IC50 = 961 nM T09572 C2OH0S 44417956 IC50 = 5 nM T09572 COA19M 44417957 IC50 = 5 nM T09572 CDF0V4 44417959 EC50 = 90 nM T09572 C3SVB8 44417960 Ki = 3465 nM T09572 C6HTW2 44417961 IC50 = 112 nM T09572 CF7QS3 44417962 EC50 = 160 nM T09572 C6TJL5 44417963 Ki = 497 nM T09572 C5GDU7 44417965 Ki = 4 nM T09572 CFU91G 44417966 IC50 = 0.3 nM T09572 C7JFN6 44417967 Ki = 148 nM T09572 C93GJO 44417968 IC50 = 313 nM T09572 CH6F8D 44417969 Ki = 228 nM T09572 CM2YT3 44417970 IC50 = 1814 nM T09572 C9RKO4 44417971 IC50 = 512 nM T09572 CNVM62 44417972 IC50 = 952 nM T09572 CF91YW 44417973 IC50 = 13 nM T09572 C3C5PN 44417974 IC50 = 212 nM T09572 CE3Q5V 44417975 IC50 = 210 nM T09572 CDT71X 44417976 IC50 = 88 nM T09572 CH2RQ7 44417977 IC50 = 243 nM T09572 C2JM1K 44417979 IC50 = 18.5 nM T09572 C6K9JW 44417981 IC50 = 904 nM T09572 C6D2EQ 44417982 IC50 = 240 nM T09572 CFU0Y7 44417983 IC50 = 1034 nM T09572 CJZ82I 44417984 Ki = 570 nM T09572 CM2EL7 44417985 Ki = 890 nM T09572 CY2I0A 44417986 IC50 = 311 nM T09572 CTYW15 44417987 Ki = 625 nM T09572 C07FSQ 44417988 IC50 = 443 nM T09572 CG63SF 44417989 Ki = 260 nM T09572 CLS47Q 44417991 IC50 = 172 nM T09572 CM4VL9 44417992 EC50 = 300 nM T09572 C7CP8I 44417993 Ki = 118 nM T09572 C8OZD0 44417994 IC50 = 122 nM T09572 CNR9E4 44417995 IC50 = 26 nM T09572 C2GZ9T 44417996 IC50 = 1100 nM T09572 CE0FS4 44417998 EC50 = 150 nM T09572 CQ3LS1 44417999 EC50 = 340 nM T09572 CWR70L 44418000 Ki = 99 nM T09572 CRP5I2 44418002 IC50 = 4 nM T09572 CP7YV8 44418003 EC50 = 904 nM T09572 C6Q7ZM 44418004 Ki = 129 nM T09572 CF4E1N 44418005 IC50 = 78 nM T09572 C8BH6G 44418006 IC50 = 1008 nM T09572 CFUG30 44418008 IC50 = 490 nM T09572 C8DIV9 44418009 IC50 = 36 nM T09572 CRO92C 44418010 IC50 = 40 nM T09572 CE51ZC 44424061 Ki = 16 nM T09572 CU78DE 44424062 Ki = 10 nM T09572 C5OXM1 44424063 Ki = 12 nM T09572 CR6TA2 44424064 Ki = 19 nM T09572 CEIA14 44424065 Ki = 194 nM T09572 CA2D9R 44424066 Ki = 4 nM T09572 CO26JC 44424067 IC50 = 38 nM T09572 CINY58 44424068 Ki = 374 nM T09572 C41UFQ 44424069 Ki = 19 nM T09572 C5THN9 44424070 IC50 = 3 nM T09572 C0G2QJ 44424071 Ki = 25 nM T09572 CLAW52 44424072 Ki = 2000 nM T09572 CUL09D 44424073 Ki = 1200 nM T09572 C7O9PT 44424166 Ki = 132 nM T09572 C8MJ5Y 44424167 Ki = 1884 nM T09572 C7GS8T 44424168 Ki = 20 nM T09572 COD05N 44424169 Ki = 373 nM T09572 C6Y3NT 44424170 Ki = 54 nM T09572 C1V5YS 44424171 Ki = 15 nM T09572 COU9D8 44424172 Ki = 20 nM T09572 CSU96B 44424173 Ki = 48 nM T09572 CZ48SF 44424174 Ki = 134 nM T09572 CA2TK3 44424175 Ki = 539 nM T09572 C4DSJ0 44424176 Ki = 2213 nM T09572 CR2GP1 44424177 Ki = 16 nM T09572 CWJ41D 44424178 Ki = 23 nM T09572 C9IC7X 44424179 Ki = 15 nM T09572 C51PEO 44424180 Ki = 7 nM T09572 CA76NC 44424181 Ki = 15 nM T09572 CP4H0T 44424182 Ki = 15 nM T09572 CKE61I 44424183 Ki = 22 nM T09572 CW8NM4 44424184 Ki = 53 nM T09572 CZ6LD4 44424185 Ki = 15 nM T09572 CSA9H2 44424186 Ki = 11 nM T09572 C9AP8V 44424187 Ki = 5 nM T09572 C7R3WV 44424188 Ki = 2.7 nM T09572 CQ6Z7X 44424189 Ki = 5.7 nM T09572 CP2W3Y 44424190 Ki = 2.1 nM T09572 CEHP70 44424191 Ki = 6 nM T09572 CBAW19 44424192 Ki = 7.6 nM T09572 CV48KH 44424193 Ki = 4.5 nM T09572 CO7A5C 44424194 Ki = 2.8 nM T09572 C7L0KT 44424195 Ki = 10.4 nM T09572 C36ROD 44424196 Ki = 2 nM T09572 CH1Z3R 44424197 Ki = 60 nM T09572 C3PMT9 44424198 Ki = 34 nM T09572 CK5ZM9 44424199 Ki = 27 nM T09572 CM5UV2 44424200 Ki = 92 nM T09572 COHK30 44424201 Ki = 92 nM T09572 CJ1S6F 44424202 Ki = 7.8 nM T09572 CPI5B7 44424203 Ki = 142 nM T09572 C59RHN 44424204 Ki = 34 nM T09572 CC7PE6 44424205 Ki = 48 nM T09572 CC45EG 44424206 Ki = 4.1 nM T09572 CNDW09 44424207 Ki = 29 nM T09572 CVKE34 44424208 Ki = 8.7 nM T09572 C5EMG3 44424209 Ki = 9.4 nM T09572 CAG2L4 44424210 Ki = 5.2 nM T09572 C04VIZ 44424211 Ki = 12 nM T09572 C51ZVB 44424212 Ki = 1.6 nM T09572 C08JMU 44424213 Ki = 1.6 nM T09572 CDB0G8 44424214 Ki = 10 nM T09572 CX21FM 44424215 Ki = 1.9 nM T09572 C8B2SV 44424216 Ki = 4.4 nM T09572 CCVG85 44424217 Ki = 11 nM T09572 CGA81M 44424218 Ki = 1.2 nM T09572 C25WLJ 44424224 Ki = 8.7 nM T09572 C5SM3Y 44424225 Ki = 181 nM T09572 C4FET2 44424228 Ki = 312 nM T09572 CBQ6F5 44424229 Ki = 7.2 nM T09572 CC4J1W 44424231 Ki = 5.4 nM T09572 CJ15CH 44424232 Ki = 21 nM T09572 C28AFI 44424233 Ki = 26 nM T09572 CC1KS2 44424234 Ki = 9.7 nM T09572 C4TDJ7 44424235 Ki = 80 nM T09572 C3PLC4 44424236 Ki = 211 nM T09572 CP90FZ 44424237 Ki = 295 nM T09572 CH2R7W 44424238 Ki = 559 nM T09572 C8BT1N 44424244 Ki = 2.3 nM T09572 CVJ2L5 44424246 Ki = 18 nM T09572 C9P1QG 44424247 Ki = 31 nM T09572 CR9L4I 44424249 Ki = 21 nM T09572 C45NIL 44424250 Ki = 54 nM T09572 CNB09T 44424252 Ki = 46 nM T09572 C2IMP0 44424253 Ki = 13 nM T09572 CW9ZC2 44424254 Ki = 9.9 nM T09572 C6OW2Z 44424255 Ki = 15 nM T09572 C4GSN5 44424256 Ki = 2.4 nM T09572 CO86IG 44424258 Ki = 3.3 nM T09572 C5F8PY 44424259 Ki = 8.9 nM T09572 C7BW3R 44424260 Ki = 146.89 nM T09572 C13AXK 44424261 Ki = 30 nM T09572 C7V2AY 44424262 Ki = 1969 nM T09572 CH17YP 44424263 Ki = 116.95 nM T09572 CW53QE 44424265 Ki = 51 nM T09572 C47BAF 44424266 Ki = 316 nM T09572 C32PLE 44424267 Ki = 85 nM T09572 C63AUS 44424268 Ki = 31 nM T09572 C1D8YR 44424269 Ki = 4.2 nM T09572 CJ25WE 44424270 Ki = 57 nM T09572 C89EXO 44425789 Ki = 50 nM T09572 C89LGK 44425790 Ki = 2100 nM T09572 CG3MY4 44425792 Ki = 1100 nM T09572 C1N0EW 44425793 Ki = 200 nM T09572 CN2I8O 44425794 Ki = 340 nM T09572 C7LMS4 44425795 Ki = 115 nM T09572 CH02JZ 44425796 Ki = 150 nM T09572 COX87N 44425797 Ki = 400 nM T09572 C89PUR 44425798 Ki = 25 nM T09572 CUP51V 44425799 Ki = 340 nM T09572 C3N2GM 44425800 Ki = 300 nM T09572 C2AE6C 44425801 Ki = 1500 nM T09572 CH04WE 44425802 Ki = 89 nM T09572 C9D4LQ 44425803 Ki = 44 nM T09572 C3REX2 44425804 Ki = 330 nM T09572 C4L5ZP 44425805 Ki = 640 nM T09572 CK7T3L 44425806 Ki = 315 nM T09572 CT1N9U 44425807 Ki = 20 nM T09572 C52ZIS 44425809 Ki = 13 nM T09572 CU7YW1 44425810 Ki = 10 nM T09572 C0WVT1 44425811 Ki = 8 nM T09572 C46FWV 44425812 Ki = 230 nM T09572 CYR4W7 44425814 Ki = 9300 nM T09572 CP1ZY6 44425815 Ki > 10000 nM T09572 CE3A2G 44425817 Ki = 20 nM T09572 CCV7H3 44425818 Ki = 210 nM T09572 C6JY8V 44425820 Ki = 620 nM T09572 CNV50P 44425821 Ki = 150 nM T09572 CA4KO2 44425822 Ki = 8000 nM T09572 C3KP5U 44425823 Ki = 2900 nM T09572 CX7TS1 44425824 Ki = 92 nM T09572 C7IF1X 44425825 Ki = 19 nM T09572 CWZ4G7 44425826 Ki = 280 nM T09572 CE2R3N 44425827 Ki = 180 nM T09572 CADK60 44425828 Ki = 100 nM T09572 CNFI93 44425830 Ki = 84 nM T09572 CY5HW2 44425832 Ki = 12 nM T09572 CKJ03V 44425834 IC50 = 5 nM T09572 CYJ20S 44425835 Ki = 6 nM T09572 C1IVD0 44425837 Ki = 45 nM T09572 CXPO87 44425839 Ki = 6 nM T09572 CBMT90 44430452 Ki = 17 nM T09572 CODL74 44430453 Ki = 6 nM T09572 CAE2N5 44430455 Ki = 5 nM T09572 CMKP65 44430458 Ki = 1 nM T09572 C8OQV2 44430459 Ki = 4 nM T09572 CNW86X 44430460 Ki = 2 nM T09572 C62BSV 44430463 Ki = 3 nM T09572 CB97TH 44430465 Ki = 50 nM T09572 CW01JX 44430468 Ki = 4 nM T09572 CU6I1H 44430471 Ki = 4 nM T09572 CJ9C8U 44430475 Ki = 3 nM T09572 C12TLF 44430476 Ki = 7 nM T09572 CQ59YW 44430477 Ki = 7 nM T09572 CH38CM 44430478 Ki = 17 nM T09572 CT37LP 44430479 Ki = 80 nM T09572 CZ8WO4 44430480 Ki = 69 nM T09572 C1UMX3 44430481 Ki = 154 nM T09572 CP6U2S 44430482 Ki = 15 nM T09572 C5YQ3O 44430483 Ki = 5 nM T09572 C2OT9F 44430484 Ki = 49 nM T09572 C7TEZ2 44430485 Ki = 17 nM T09572 C8J0LH 44430486 Ki = 39 nM T09572 CX1D3I 44430487 Ki = 21 nM T09572 C5K1DQ 44430488 Ki = 46 nM T09572 CRT5O9 44430489 Ki = 26 nM T09572 CAG1M5 44430490 Ki = 143 nM T09572 CX03CA 44430493 Ki = 14 nM T09572 CTM7G1 44430494 Ki = 8 nM T09572 CTK8S7 44430495 Ki = 70 nM T09572 CIG9Y6 44430496 Ki = 19 nM T09572 CR5EU8 44430498 Ki = 18 nM T09572 CX81ZL 44430499 Ki = 28 nM T09572 CKOL19 44430500 Ki = 14 nM T09572 C09UFN 44430501 Ki = 45 nM T09572 CJ81UG 44434143 Ki = 22 nM T09572 C15TRQ 44434144 Ki = 431 nM T09572 C16UDV 44434145 Ki = 99 nM T09572 CC03AH 44434146 Ki = 45 nM T09572 C5H1MB 44434148 Ki = 17 nM T09572 CYNE36 44434149 Ki = 19 nM T09572 CVFM10 44434151 Ki = 13.1 nM T09572 CA98YS 44434152 Ki = 73 nM T09572 CN80KD 44434153 Ki = 117 nM T09572 CM6LD3 44434154 Ki = 6.1 nM T09572 CY45FT 44434155 Ki = 171 nM T09572 CZ18JV 44434156 Ki = 4 nM T09572 C7LD6V 44437494 Ki = 543.25 nM T09572 C1I2BU 44437495 Ki = 1445.44 nM T09572 CS9UQ1 44437496 Ki = 425 nM T09572 C4SV8L 44437497 Ki = 186 nM T09572 CO8DT9 44437498 Ki = 2640 nM T09572 C9R8WN 44437499 Ki = 5860 nM T09572 C3ZDU4 44437500 Ki > 1000 nM T09572 CP36JI 44437501 Ki = 6025.6 nM T09572 CCMV89 44437514 Ki = 6380 nM T09572 CO20QU 44437515 Ki > 1000 nM T09572 CRD6O8 44437516 Ki = 312.61 nM T09572 CW09ML 44437517 Ki = 273 nM T09572 CE5OX7 44437518 Ki > 1000 nM T09572 CXH06Q 44437519 Ki = 509 nM T09572 CYK2O7 44437520 Ki = 257.04 nM T09572 CAV9L2 44437522 Ki = 421 nM T09572 C4HZX3 44437523 Ki = 595 nM T09572 CXBE83 44437524 Ki = 214.78 nM T09572 C4X0AD 44437525 Ki = 254 nM T09572 CPLN85 44437526 Ki = 947 nM T09572 CTKX20 44437528 Ki = 213.8 nM T09572 CE08HO 44437541 Ki = 169.82 nM T09572 C7VBE4 44437542 Ki = 1200 nM T09572 CV6S2Q 44437544 Ki = 1080 nM T09572 CYC56F 44437547 Ki = 388 nM T09572 CPDS73 44437553 Ki = 96.6 nM T09572 CZ9L4F 44437555 Ki = 204 nM T09572 C1AU2N 44437557 Ki = 251 nM T09572 C61UVK 44437558 Ki = 144 nM T09572 C0IQ8W 44437609 Ki = 149 nM T09572 CBG34A 44437612 Ki = 143 nM T09572 CC1L2V 44437614 Ki = 165.96 nM T09572 CJQ1X5 44437620 Ki = 769 nM T09572 CS3GI1 44437622 Ki = 173 nM T09572 CEB9V8 44438737 IC50 > 2000 nM T09572 CJ79PE 44438739 IC50 = 1520 nM T09572 C9T7JL 44438740 IC50 = 773 nM T09572 CB9S3W 44438741 IC50 = 165 nM T09572 CL20OD 44438742 IC50 = 64 nM T09572 C71UWM 44438745 IC50 = 4010 nM T09572 CBJ5R9 44438747 IC50 = 31 nM T09572 C5VFD8 44438748 IC50 = 15 nM T09572 CW8GU6 44438753 IC50 = 86 nM T09572 CS9D3H 44438755 IC50 = 26 nM T09572 C65EMO 44440586 Ki = 260 nM T09572 C6FGD1 44440587 Ki = 101 nM T09572 C8ZA4N 44440588 Ki = 1090 nM T09572 CZ1L5J 44440593 Ki = 1000 nM T09572 C9IBX4 44440599 Ki = 176 nM T09572 C0NBF9 44442050 IC50 = 3590 nM T09572 CUC4A6 44442051 IC50 > 33000 nM T09572 C7EH8P 44442053 IC50 = 3 nM T09572 C8EAD0 44442054 IC50 = 411 nM T09572 C03OKE 44442056 IC50 = 5010 nM T09572 C9BKO7 44442058 IC50 = 106 nM T09572 CZVQ72 44442059 IC50 = 119 nM T09572 CBTV83 44442060 IC50 = 2990 nM T09572 CW41ZF 44442061 IC50 = 2300 nM T09572 C23MNK 44442062 IC50 = 2130 nM T09572 C1PEQ4 44442063 IC50 = 68 nM T09572 CANQ03 44442064 IC50 = 7 nM T09572 CC6S0I 44442065 IC50 = 25 nM T09572 CXJ52D 44442066 IC50 = 571 nM T09572 CD5G2R 44442067 IC50 = 847 nM T09572 CE0Y1I 44442068 IC50 = 2520 nM T09572 CO3V4T 44442069 IC50 = 4800 nM T09572 C4CRF6 44442070 IC50 = 9920 nM T09572 CE52RC 44442071 IC50 = 97 nM T09572 C2A0OM 44442090 IC50 = 8 nM T09572 CX5J6I 44442093 IC50 = 231 nM T09572 C10KDT 44442095 IC50 = 0.1 nM T09572 CR3KI9 44442097 IC50 = 54 nM T09572 CE4LG3 44442098 IC50 = 1390 nM T09572 CLU51Z 44442100 IC50 = 5100 nM T09572 C06WTB 44442118 IC50 = 22 nM T09572 CPW23O 44442119 IC50 = 89 nM T09572 CT3N0B 44442120 IC50 = 13 nM T09572 C8VEW9 44442121 IC50 = 28 nM T09572 C2Y1XP 44442124 IC50 = 61 nM T09572 CK57FP 44442130 IC50 = 58 nM T09572 CGLN40 44442134 IC50 = 16 nM T09572 C13TNE 44442135 IC50 = 50 nM T09572 C2FAQ7 44442139 IC50 = 9 nM T09572 CBN4Q3 44442144 IC50 = 35 nM T09572 CSQN12 44442148 IC50 = 80 nM T09572 C0SMR6 44442151 IC50 = 33 nM T09572 CBV07Y 44442153 IC50 = 20 nM T09572 C4Z8HF 44442156 IC50 = 39 nM T09572 CV3ZI1 44454966 Ki = 25 nM T09572 CU8EX2 44455336 Ki = 0.5 nM T09572 COU5A6 44455367 Ki = 47 nM T09572 C7B1KA 44455368 Ki = 10 nM T09572 CQKH50 44455414 Ki = 5 nM T09572 CK4O6B 44455417 Ki = 20 nM T09572 C0I6SN 44455443 Ki = 31 nM T09572 CRN57M 44455444 Ki = 5.2 nM T09572 CQ0WM7 44469273 IC50 = 2.6 nM T09572 CNW41S 44539369 Ki = 2920 nM T09572 CJE2Q6 44555375 IC50 = 1.2 nM T09572 C4LJ6X 44557554 IC50 = 19 nM T09572 C2X1BC 44562403 IC50 = 804 nM T09572 CK2GC9 44562404 IC50 = 104 nM T09572 C21KTW 44562405 IC50 = 903 nM T09572 COQ7L5 44562415 IC50 = 82 nM T09572 CX39BW 44562416 IC50 = 2340 nM T09572 CZVN14 44562441 IC50 > 33000 nM T09572 C7C5GX 44562442 IC50 = 43 nM T09572 C6X1CW 44562443 IC50 = 9650 nM T09572 CC57QH 44562461 IC50 = 1500 nM T09572 CZT5U2 44562462 IC50 = 927 nM T09572 CTV75H 44562479 IC50 = 347 nM T09572 CHN81A 44562480 IC50 = 2140 nM T09572 CCY92R 44562481 IC50 = 636 nM T09572 C4WAK1 44562499 IC50 = 3050 nM T09572 CH40TM 44562500 IC50 = 29 nM T09572 C1NG5P 44562501 IC50 = 111 nM T09572 C4IK2N 44562521 IC50 = 2260 nM T09572 CP80OG 44562522 IC50 = 104 nM T09572 CE5M8W 44562523 IC50 = 1250 nM T09572 CK6PR8 44562524 IC50 = 169 nM T09572 C9QW4M 44562542 IC50 = 313 nM T09572 CYDB09 44562543 IC50 = 303 nM T09572 C6USZ1 44562544 IC50 = 269 nM T09572 CEJ3G1 44562545 IC50 = 122 nM T09572 C59XKS 44562562 IC50 = 113 nM T09572 CAPH48 44562563 IC50 = 58 nM T09572 C9XD5G 44562564 IC50 = 67 nM T09572 CJB05V 44562565 IC50 = 66 nM T09572 C1SUW5 44562600 IC50 = 71 nM T09572 C81IMZ 44573820 IC50 = 9.6 nM T09572 CEF6J8 44573821 IC50 = 2.1 nM T09572 CT2FW6 44573822 IC50 = 2.1 nM T09572 C4I5UB 44573823 IC50 = 19 nM T09572 CXWQ34 44573931 IC50 = 1.7 nM T09572 C6U0EY 44573932 IC50 = 9.9 nM T09572 C04SIR 44573964 IC50 = 125 nM T09572 CAT49R 44574008 IC50 = 0.15 nM T09572 C0VQ8Y 44574357 IC50 = 54 nM T09572 CQZ1Y2 44574358 IC50 = 42 nM T09572 C0SOD6 44574359 IC50 = 42 nM T09572 C95TVW 44592169 Ki = 3.16 nM T09572 COR08L 44592214 Ki = 3.3 nM T09572 CO0RY5 44592215 Ki = 3 nM T09572 CO6X8L 44592256 IC50 = 83.18 nM T09572 CO6ES5 44592257 IC50 = 104.71 nM T09572 CD06ZV 45178545 IC50 = 18000 nM T09572 C3BWP6 45266975 Ki = 1413 nM T09572 CJVC17 45266979 Ki = 30 nM T09572 CP1UX8 45267015 Ki = 3473 nM T09572 C1N5ZL 45267385 IC50 = 55 nM T09572 C4AZD3 45267386 IC50 = 444 nM T09572 C8LPF5 45267399 IC50 = 597 nM T09572 C8PR5X 45267430 IC50 = 21 nM T09572 C17EPN 45267561 IC50 = 83 nM T09572 CA4ZJ2 45267565 IC50 = 260 nM T09572 CNZ95W 45267576 IC50 = 100 nM T09572 CVPT19 45267577 IC50 = 5.4 nM T09572 C7SJ4A 45267654 IC50 = 300 nM T09572 CM23AU 45267709 IC50 = 196 nM T09572 CGB32I 45267714 IC50 = 21 nM T09572 CO3Y0N 45267724 IC50 = 120 nM T09572 CI7KZ2 45267735 IC50 = 17 nM T09572 CC5OP0 45267739 IC50 = 27 nM T09572 CXJ8H3 45267746 IC50 = 152 nM T09572 CCS2E7 45267809 Ki = 17380 nM T09572 CV4W6Y 45267812 Ki = 1951 nM T09572 CZ8G9K 45267814 Ki = 4560 nM T09572 C37UGL 45267827 Ki = 149 nM T09572 CH4V7J 45267849 IC50 = 11765 nM T09572 CP85WO 45268247 IC50 = 71 nM T09572 CW5C8M 45268457 IC50 = 320 nM T09572 C4G1SL 45268465 IC50 = 48 nM T09572 C84UTO 45268470 IC50 = 4 nM T09572 COZ7J8 45268527 IC50 = 130 nM T09572 C7VZR5 45268637 IC50 = 112 nM T09572 CV1IR5 45268644 IC50 = 412 nM T09572 CXSQ09 45268694 Ki = 2334 nM T09572 CJFQ65 45268721 Ki = 5642 nM T09572 CGL25F 45268725 Ki = 3567 nM T09572 CPH10U 45269335 IC50 = 102 nM T09572 C63KED 45269336 IC50 = 44 nM T09572 CHR31D 45269555 Ki = 5114 nM T09572 CA3MZ6 45269996 IC50 = 417 nM T09572 C5DIS2 45270014 IC50 = 5 nM T09572 CF0DL4 45270139 IC50 = 35 nM T09572 CC14UH 45270147 IC50 = 330 nM T09572 C2UNR9 45270157 IC50 = 160 nM T09572 CPG7D6 45270273 IC50 = 617 nM T09572 C0J6BO 45270297 IC50 = 138 nM T09572 C23PMF 45270302 IC50 = 125 nM T09572 C9WNG1 45270303 IC50 = 46 nM T09572 C4SXQ3 45270319 IC50 = 66 nM T09572 C26DVR 45270386 Ki = 2056 nM T09572 C7LW6A 45270392 Ki = 5 nM T09572 CL71EJ 45270393 Ki = 312 nM T09572 CKLX79 45270416 IC50 = 1800 nM T09572 C3A0NB 45270802 IC50 = 4 nM T09572 C35TNH 45270803 IC50 = 150 nM T09572 C3GLV8 45270841 IC50 = 28 nM T09572 CD5OS6 45270850 IC50 = 67 nM T09572 C42GYR 45271095 IC50 = 13 nM T09572 C1F5RT 45271103 IC50 = 236 nM T09572 CCN0F4 45271111 IC50 = 40 nM T09572 CS9M8B 45271114 IC50 = 36 nM T09572 CY70FL 45271134 IC50 = 10 nM T09572 C5YL6K 45271219 Ki = 105 nM T09572 C97WCQ 45271221 Ki = 1078 nM T09572 CR3S4Z 45271246 Ki = 13890 nM T09572 CO04UR 45271549 IC50 = 145 nM T09572 C13PCQ 45271633 IC50 = 8 nM T09572 C3OA8C 45271642 IC50 = 30 nM T09572 CP7CX1 45271647 IC50 = 142 nM T09572 CH1PS3 45271663 IC50 = 173 nM T09572 CM4ZX1 45271673 IC50 = 17 nM T09572 CJN52K 45271829 IC50 = 26 nM T09572 CF9L1B 45271839 IC50 = 4.8 nM T09572 CIWH57 45271907 IC50 = 7.1 nM T09572 C12DAS 45271908 IC50 = 11 nM T09572 C36SRE 45271994 IC50 = 81.8 nM T09572 C73LNM 45272006 IC50 = 111 nM T09572 CMYT82 45272014 IC50 = 23 nM T09572 C60DPZ 45272024 IC50 = 82 nM T09572 C2MKZ1 45272040 IC50 = 308 nM T09572 CWD50J 45272111 Ki = 15606 nM T09572 C7O1UV 45272117 Ki = 4678 nM T09572 C5CEH0 45272120 Ki = 133 nM T09572 C6FCW0 45272539 IC50 = 66 nM T09572 CKI1W9 45272701 IC50 = 8.2 nM T09572 CJ52PS 45272816 IC50 = 49 nM T09572 CD6FR7 45272837 IC50 = 57 nM T09572 C3GUS5 45272853 IC50 = 38 nM T09572 C2YI4R 45272942 Ki = 2584 nM T09572 CY65HN 45272944 Ki = 36588 nM T09572 C3F7SQ 45272984 Ki = 4135 nM T09572 C7QZG5 45272985 Ki = 9332 nM T09572 CYD3P4 45273335 IC50 = 0.87 nM T09572 C9JQT2 45273392 IC50 = 815 nM T09572 CPTE06 45273401 IC50 = 40 nM T09572 CG4YS2 45273406 IC50 = 144 nM T09572 CZ7R6G 45273623 IC50 = 30 nM T09572 C2K6RW 45273638 IC50 = 140 nM T09572 C2AB8E 45273642 IC50 = 122 nM T09572 CSGK15 45273659 IC50 = 61 nM T09572 CKM6P4 45273703 IC50 = 4.6 nM T09572 CLFN69 45273777 IC50 = 28 nM T09572 CP7OZ1 45273778 IC50 = 90 nM T09572 COD72W 45273783 IC50 = 63 nM T09572 CCJR41 45273790 IC50 = 63 nM T09572 C3TZ8X 45273801 IC50 = 19 nM T09572 CX9T5I 45273802 IC50 = 11 nM T09572 CX9LC1 45273887 IC50 = 3057 nM T09572 C2GKC7 45278576 Ki = 124 nM T09572 C81XVO 45278577 Ki = 17 nM T09572 CVD12N 45278578 Ki = 13 nM T09572 CY9SZ3 45278579 Ki = 0.7 nM T09572 CPT17U 45278657 Ki = 76 nM T09572 CQ4J0K 45278977 Ki = 26 nM T09572 C79CHB 45279061 Ki = 3.4 nM T09572 C35VWA 45279062 Ki = 6.5 nM T09572 CH3YM7 45279064 Ki = 6.5 nM T09572 C9GZ5B 45279148 Ki = 2.4 nM T09572 C6DU8B 45279233 Ki = 9 nM T09572 CT30ZQ 45279319 Ki = 28 nM T09572 CJ20EF 45279321 Ki = 15 nM T09572 CE7WZ3 45279402 Ki = 2.3 nM T09572 C8XY6M 45279488 Ki = 21 nM T09572 C0Y2PW 45279489 Ki = 3.5 nM T09572 C7DXG1 45279490 Ki = 0.5 nM T09572 CER6A7 45279491 Ki = 86 nM T09572 C2K8NV 45279493 Ki = 4.4 nM T09572 CX01LN 45279583 Ki = 4.8 nM T09572 CR0N4Z 45279585 Ki = 0.4 nM T09572 C7XI9W 45279680 Ki = 12 nM T09572 C84XIH 45279772 Ki = 15 nM T09572 CZF27R 45279773 Ki = 5.3 nM T09572 C58PTY 45279868 Ki = 3.1 nM T09572 CJO30G 45279869 Ki = 0.8 nM T09572 CL0D6F 45279871 Ki = 13 nM T09572 CYUP42 45279872 Ki = 9.1 nM T09572 CWM86N 45484974 IC50 = 46 nM T09572 CN1OK5 45484984 IC50 = 210 nM T09572 CGLF37 45484995 IC50 = 120 nM T09572 C4X8LF 45485002 IC50 = 26 nM T09572 CQL2O6 45485003 IC50 = 81 nM T09572 C3NFA0 45485004 IC50 = 200 nM T09572 CIX49Y 45485018 IC50 = 230 nM T09572 CHWT32 45485028 IC50 = 7.6 nM T09572 CI97CR 45485029 IC50 = 100 nM T09572 CBZ02X 45485038 IC50 = 64 nM T09572 C7GQ2P 45485043 IC50 = 600 nM T09572 CGOS24 45485061 IC50 = 8 nM T09572 CLX9C8 45485062 IC50 = 2.9 nM T09572 C9JG7Q 45485063 IC50 = 4 nM T09572 C53PKX 45485077 IC50 = 9.6 nM T09572 CREA46 45487283 IC50 = 3.5 nM T09572 C04UFC 45487284 IC50 = 4.4 nM T09572 C7PF5S 45487309 IC50 = 3.5 nM T09572 CTCP93 45487326 IC50 > 1000 nM T09572 CXS6B7 45487330 IC50 = 29 nM T09572 C8ZP0F 45487331 IC50 = 5.4 nM T09572 CF8J3Q 45487356 IC50 = 11 nM T09572 C6KSR1 45487366 IC50 = 30 nM T09572 CSI8X4 45487371 IC50 > 1000 nM T09572 C6FVJ7 45487372 IC50 = 5 nM T09572 C1SEH5 45487375 IC50 > 1000 nM T09572 C1AM2G 45487382 IC50 = 5.9 nM T09572 CC1SO0 45487383 IC50 = 3.3 nM T09572 C3QU2C 45487384 IC50 = 7 nM T09572 COF5G1 45487385 IC50 = 11 nM T09572 C7LQ4D 45487390 IC50 = 5.2 nM T09572 CAB4D7 45487391 IC50 = 4.9 nM T09572 CK9I3H 45487392 IC50 = 34 nM T09572 CMX27T 45487640 IC50 = 2.6 nM T09572 C5NO1K 45487641 IC50 = 45 nM T09572 CR10DI 45487647 IC50 = 1.4 nM T09572 CS17WK 45487652 IC50 = 3.5 nM T09572 CAQ2D8 45487653 IC50 = 6.8 nM T09572 C3A7QW 45487657 IC50 = 4.6 nM T09572 CB9K2G 45487660 IC50 = 1.3 nM T09572 CJ8R3S 45487668 IC50 = 0.22 nM T09572 CN1V0Y 45487671 IC50 = 0.12 nM T09572 CWH0O7 45487673 IC50 = 6.3 nM T09572 CCZR81 45487674 IC50 = 0.35 nM T09572 CTB2P0 46188603 IC50 = 241 nM T09572 C3UN9A 46188959 IC50 = 1173 nM T09572 CS6P3L 46878210 Ki = 338 nM T09572 C07TYF 46899578 IC50 = 1750 nM T09572 C4D0HN 46899579 IC50 = 450 nM T09572 CYSC07 46899581 IC50 = 540 nM T09572 CI05ZH 46899582 IC50 = 1160 nM T09572 C7JP6X 46902024 IC50 = 120 nM T09572 CS46RV 46902025 IC50 = 1660 nM T09572 C08OLW 46902026 IC50 = 920 nM T09572 CHU2O6 46933537 IC50 = 2 nM T09572 C9YZ5I 46933538 IC50 = 0.6 nM T09572 C8A0LD 49801837 IC50 = 23 nM T09572 CG3VX4 49865653 IC50 = 45 nM T09572 CMHY97 49865654 IC50 = 21 nM T09572 C9I0SK 49865678 IC50 = 68 nM T09572 CE09ML 49865679 IC50 = 71 nM T09572 CH5WD6 49865680 IC50 = 35 nM T09572 C9OKI3 49865708 IC50 = 269 nM T09572 CT98KS 49865738 IC50 = 600 nM T09572 CGXO13 49865739 IC50 = 35 nM T09572 C0V2OU 49865789 IC50 = 140 nM T09572 CZ9H6T 49865790 IC50 = 261 nM T09572 CC6B0N 49865868 IC50 = 110 nM T09572 C7Z5TE 49865869 IC50 = 528 nM T09572 C7OF6U 49865870 IC50 = 1620 nM T09572 CI52NU 49865871 IC50 = 87 nM T09572 C5TN3P 49865927 IC50 = 10 nM T09572 CBJ87H 49865928 IC50 = 15 nM T09572 CPHK47 49865929 IC50 = 112 nM T09572 CROD23 49865975 IC50 = 646 nM T09572 C15SMZ 49865976 IC50 = 88 nM T09572 C3G6MD 49865977 IC50 = 336 nM T09572 CBW0I6 49866034 IC50 = 1450 nM T09572 CIP9U4 49866035 IC50 = 13 nM T09572 CS8OU5 49866036 IC50 = 37 nM T09572 C3HI5E 49866086 IC50 = 678 nM T09572 C4PR5M 49866087 IC50 = 566 nM T09572 CEA02K 49866088 IC50 = 9 nM T09572 CK6AX0 49866089 IC50 = 106 nM T09572 C1N4YP 50908737 Ki = 4.9 nM T09572 C3SJ6Y 50908738 Ki = 2.6 nM T09572 C92GDH 50908739 Ki = 2.4 nM T09572 CIRP71 52917998 IC50 = 7 nM T09572 CT0B1S 52917999 IC50 = 12 nM T09572 CFX76G 52918016 IC50 = 12 nM T09572 C47RHB 52918017 IC50 = 27 nM T09572 C9SE1W 52940981 Ki = 33.96 nM T09572 CV8Q3Y 52941054 Ki = 20 nM T09572 C4NUM9 52941152 Ki = 14 nM T09572 CH4X0U 52941195 Ki = 14 nM T09572 CW6CG4 52941272 Ki = 20.99 nM T09572 CFI49B 52941492 Ki = 16 nM T09572 C1HS4J 52941518 Ki = 8.71 nM T09572 CUV8I6 52941526 Ki = 37.7 nM T09572 C9NX0A 52941539 Ki = 7.6 nM T09572 CZM85N 52941615 Ki = 11 nM T09572 CMN74I 52941621 Ki = 8.4 nM T09572 C1YLX8 52941699 Ki = 5.2 nM T09572 C34WMT 52942456 Ki = 3.8 nM T09572 CAH6F7 52942539 Ki = 4.977 nM T09572 CQ20HZ 52942540 Ki = 15 nM T09572 CJOB30 52942547 Ki = 5.2 nM T09572 CIN1J9 52942550 Ki = 62 nM T09572 C79HTE 52942685 Ki = 2.799 nM T09572 CXK65J 52942795 Ki = 11 nM T09572 CT8UE5 52942796 Ki = 5.6 nM T09572 C13YUX 52942885 Ki = 1.901 nM T09572 CXYD26 52943353 Ki = 21.98 nM T09572 C6BZO9 52943420 Ki = 5.395 nM T09572 C2GR9I 52943485 Ki = 28.97 nM T09572 CWX75K 52943587 Ki = 8.892 nM T09572 C0SML4 52943689 Ki = 47.97 nM T09572 CFTH05 52943690 Ki = 59.98 nM T09572 CD3H8P 52943712 Ki = 295.12 nM T09572 CX2RY7 52943873 Ki = 1.6 nM T09572 C8R4JF 52943912 Ki = 23.01 nM T09572 CE0MV7 52943913 Ki = 15 nM T09572 C3GQC4 52943978 Ki = 15 nM T09572 CE84SY 52944068 Ki = 708 nM T09572 C2U4VH 52944540 Ki = 181.13 nM T09572 C0U8RC 52944577 Ki = 47.97 nM T09572 C6L3EG 52944805 Ki = 6300 nM T09572 CV9B7X 52944859 Ki = 17.99 nM T09572 CPV63Q 52944920 Ki = 46.03 nM T09572 C0C2TV 52944948 Ki = 92.04 nM T09572 CEB4J0 52944997 Ki = 7.8 nM T09572 C5DCJ2 52945048 Ki = 2.099 nM T09572 CV6T4N 52945087 Ki = 1.6 nM T09572 C6HNI1 52945088 Ki = 30.97 nM T09572 CT8X7J 52945129 Ki = 10.99 nM T09572 C1MHT3 52945130 Ki = 1.199 nM T09572 CK7JS2 52945154 Ki = 15 nM T09572 CC1NT2 52945806 Ki = 7.762 nM T09572 CG8Z4H 52945863 Ki = 4.102 nM T09572 CXZI97 52946021 Ki = 133.97 nM T09572 C83GRH 52946062 Ki = 26 nM T09572 C9J6PV 52946082 Ki = 20 nM T09572 CTS78H 52946137 Ki = 33.96 nM T09572 CTF7I1 52946184 Ki = 2.698 nM T09572 C6X9RM 52946259 Ki = 5.998 nM T09572 C6HBD0 52947025 Ki = 3500 nM T09572 CK1FT4 52947054 Ki = 7.194 nM T09572 CU86TE 52947140 Ki = 132.13 nM T09572 CL6TY3 52947141 Ki = 20.99 nM T09572 C6CBM4 52947251 Ki = 14 nM T09572 CN6EW2 52947267 Ki = 53.95 nM T09572 CSJ0U6 52947270 Ki = 17 nM T09572 CW6MI3 52947297 Ki = 128 nM T09572 C8PLT3 52947314 Ki = 373.25 nM T09572 CD1P9I 52947331 Ki = 15 nM T09572 C5W8CU 52947407 Ki = 13 nM T09572 CBG8U3 52947408 Ki = 8.71 nM T09572 CXHO23 52947539 Ki = 4.498 nM T09572 C1EY0A 52947542 Ki = 4.395 nM T09572 CTS9E4 52947550 Ki > 5000 nM T09572 CAHV60 52947558 Ki = 7.6 nM T09572 CZ19DQ 52947578 Ki = 1200 nM T09572 C4UN6O 52947610 Ki = 6.998 nM T09572 CCIG41 52947616 Ki = 12.6 nM T09572 C7KTG3 52948254 Ki = 6600 nM T09572 C5M3KF 52948459 Ki > 1000 nM T09572 CRK14T 52948531 Ki = 53.95 nM T09572 CP2EZ8 52948553 Ki = 30.97 nM T09572 C03ORG 52948635 Ki = 5.702 nM T09572 CZ51UD 52948636 Ki = 3.304 nM T09572 CU6QX1 52948758 Ki = 10.4 nM T09572 C76WHV 52948835 Ki = 25 nM T09572 C7SAC6 52948857 Ki = 1.2 nM T09572 CERH05 52948916 Ki = 2.399 nM T09572 C62QLU 52948951 Ki = 9.397 nM T09572 C4EOB2 52949472 Ki = 15 nM T09572 CNG60D 52949479 Ki = 311.89 nM T09572 C25FGA 52949693 Ki = 79.98 nM T09572 C61XZN 52949768 Ki = 9.705 nM T09572 CD26UA 52949812 Ki = 26.98 nM T09572 C3N6DP 52949912 Ki = 11.99 nM T09572 CS02MO 52949941 Ki = 7.2 nM T09572 C0M7FO 52949955 Ki = 7.603 nM T09572 C94WRG 52949956 Ki = 84.92 nM T09572 CQYM81 52950112 Ki = 10.99 nM T09572 CHNX58 53317305 IC50 = 30 nM T09572 CDH87Y 53317306 IC50 = 5.9 nM T09572 CK3MZ0 53317307 IC50 = 7.7 nM T09572 CG6CM0 53317308 IC50 > 1000 nM T09572 CV9W1B 53317524 IC50 = 650 nM T09572 C13SNK 53318592 IC50 = 18 nM T09572 CGWD27 53318593 IC50 = 6.7 nM T09572 C54SRN 53318594 IC50 = 6.8 nM T09572 C74CVF 53318595 IC50 = 16 nM T09572 CK1ZI3 53318801 IC50 = 24 nM T09572 C1VDP8 53319915 IC50 > 1000 nM T09572 CWLQ84 53320117 IC50 = 23 nM T09572 CJ7RL2 53321222 IC50 = 640 nM T09572 CML70D 53321223 IC50 = 3.8 nM T09572 C4BW7G 53322554 IC50 = 12 nM T09572 C98PDX 53322555 IC50 = 4.2 nM T09572 C0HC8D 53324076 IC50 = 7 nM T09572 CHRK49 53324269 IC50 = 180 nM T09572 C6IDZ5 53325163 IC50 = 150 nM T09572 CS3L5G 53325164 IC50 = 22 nM T09572 COD2Y6 53325165 IC50 = 51 nM T09572 CX1RG6 53325166 IC50 > 1000 nM T09572 C9ZF4V 53326457 IC50 = 18 nM T09572 C1UZ8E 54579971 IC50 = 4600 nM T09572 CTA9K1 54579972 IC50 = 3120 nM T09572 C1GXF9 54579973 IC50 = 14 nM T09572 CLW26Q 54580457 IC50 = 70 nM T09572 C8W4CO 54580458 IC50 = 530 nM T09572 CTN5U4 54580459 IC50 = 1130 nM T09572 CQ8E0H 54580923 IC50 = 3180 nM T09572 CQ6V1E 54581466 IC50 = 310 nM T09572 CA2Y3W 54581468 IC50 = 100 nM T09572 C1PWI9 54581469 IC50 > 10000 nM T09572 C8NE4S 54581980 IC50 = 2600 nM T09572 CBK79N 54581986 IC50 > 10000 nM T09572 CUN59X 54582014 IC50 = 840 nM T09572 C5S1ZK 54582015 IC50 = 350 nM T09572 CL02CG 54582016 IC50 > 10000 nM T09572 CGA01C 54582476 IC50 = 360 nM T09572 C2CAO0 54582957 IC50 = 31 nM T09572 CZ3DW2 54582958 IC50 = 170 nM T09572 CM56TD 54582959 IC50 > 10000 nM T09572 CS3P4K 54582960 IC50 = 1600 nM T09572 CD0WT4 54582961 IC50 = 91 nM T09572 C72AXY 54583209 IC50 = 5380 nM T09572 C2DEZ6 54583449 IC50 > 10000 nM T09572 C1R7PQ 54583912 IC50 = 2300 nM T09572 CP0WN1 54583922 IC50 > 10000 nM T09572 CN6E9W 54583953 IC50 = 250 nM T09572 C6UED1 54583954 IC50 = 41 nM T09572 C68OSI 54584181 IC50 = 30 nM T09572 CRZY72 54584417 IC50 > 10000 nM T09572 C3VO1U 54584857 IC50 = 4800 nM T09572 CR3ON1 54584904 IC50 = 2050 nM T09572 C3C8QF 54584905 IC50 = 640 nM T09572 C0V6NH 54584906 IC50 = 2200 nM T09572 CKM78Q 54584907 IC50 > 10000 nM T09572 C7UY2T 54584908 IC50 = 150 nM T09572 CJ03KM 54585374 IC50 = 670 nM T09572 C0TC3L 54585375 IC50 = 410 nM T09572 C7PI2T 54585376 IC50 = 3800 nM T09572 CVE5B9 54585377 IC50 = 170 nM T09572 CIU2O3 54585378 IC50 = 170 nM T09572 C8JUO0 54585827 IC50 = 3200 nM T09572 C0C2BE 54585833 IC50 = 1520 nM T09572 C10GJU 54585861 IC50 = 940 nM T09572 CPX76L 54585862 IC50 = 1520 nM T09572 CW31VH 54585863 IC50 = 24 nM T09572 C2M9RO 54585864 IC50 = 30 nM T09572 CD71UB 54586089 IC50 = 50 nM T09572 CU1F9B 54586090 IC50 > 6000 nM T09572 C5K7CF 54586330 IC50 = 160 nM T09572 CM86YJ 54586331 IC50 = 1020 nM T09572 CA68VP 54586332 IC50 > 10000 nM T09572 CH15VT 54586333 IC50 > 10000 nM T09572 CLUV37 54586334 IC50 > 10000 nM T09572 CSY9Q5 54586798 IC50 > 10000 nM T09572 C3HE2I 54586826 IC50 = 2620 nM T09572 C27KZJ 54586827 IC50 > 10000 nM T09572 CI5G2O 54587365 IC50 > 10000 nM T09572 CAL94R 54587366 IC50 > 10000 nM T09572 CX74PC 54587367 IC50 > 10000 nM T09572 CI4ON9 54587368 IC50 = 140 nM T09572 C7Y3PM 56589628 IC50 = 5.6 nM T09572 CCG6D9 56597407 IC50 = 34 nM T09572 CAC5B2 56597542 IC50 = 27 nM T09572 CTK41N 56597689 IC50 = 21 nM T09572 CN54TH 56597851 IC50 = 23 nM T09572 CZNV53 56597988 IC50 = 22 nM T09572 CI6B8D 56597990 IC50 = 93 nM T09572 CSU5C1 56597991 IC50 = 25 nM T09572 CJ4V0G 56598130 IC50 = 29 nM T09572 CK6VF3 56598528 IC50 = 19 nM T09572 C5F8IX 56666754 IC50 = 9.9 nM T09572 CKQ47D 56666755 IC50 = 4.6 nM T09572 CT0JY2 56666756 IC50 = 33 nM T09572 CQO6F8 56673711 IC50 > 10000 nM T09572 C8MAJ6 56673713 IC50 = 5.5 nM T09572 C7BDU4 56673714 IC50 = 140 nM T09572 CES2I1 56680348 IC50 = 6.8 nM T09572 CYE9C0 56683679 IC50 = 50 nM T09572 C3OM0R 57390252 IC50 = 61 nM T09572 CVM2Z0 57390738 IC50 = 40 nM T09572 C4AVT1 57390739 IC50 = 91 nM T09572 CB6R2C 57391027 IC50 = 86 nM T09572 C3I2XE 57391028 IC50 = 11 nM T09572 C56RAV 57391029 IC50 > 1000 nM T09572 CCTK32 57391030 IC50 = 480 nM T09572 CZ4FY6 57391045 IC50 = 46 nM T09572 C0P1NW 57391572 IC50 = 200 nM T09572 CWL86O 57391573 IC50 = 3300 nM T09572 CBY5V0 57391574 IC50 = 180 nM T09572 CP8Y0U 57391575 IC50 > 20000 nM T09572 CVA0I2 57392546 IC50 = 14 nM T09572 CM7NG4 57392547 IC50 = 5 nM T09572 C8SEO1 57392548 IC50 = 380 nM T09572 CT06UE 57392549 IC50 = 12 nM T09572 CHOU93 57392823 IC50 = 22 nM T09572 C4VSR8 57392824 IC50 = 4.7 nM T09572 C0GK5W 57392835 IC50 = 19 nM T09572 CBX75K 57393331 IC50 = 200 nM T09572 CKW2R8 57393332 IC50 = 0.9 nM T09572 CVP38Z 57394271 IC50 = 20 nM T09572 CW8T3G 57394272 IC50 = 20 nM T09572 C2EWB0 57394273 IC50 = 423 nM T09572 CRB28X 57394274 IC50 = 7 nM T09572 C4O0AK 57394275 IC50 = 50 nM T09572 CI7J8D 57394546 IC50 > 1000 nM T09572 CX0AM8 57394547 IC50 > 1000 nM T09572 CA3YG5 57395049 IC50 = 700 nM T09572 C19CVL 57395050 IC50 = 40 nM T09572 CC64OF 57396018 IC50 = 20 nM T09572 CX6EZ4 57396019 IC50 = 30 nM T09572 C39VRQ 57396020 IC50 = 50 nM T09572 C74WKY 57396021 IC50 = 34 nM T09572 C8IU0W 57396022 IC50 = 27 nM T09572 CV26IT 57396293 IC50 = 1200 nM T09572 CWY6C2 57396294 IC50 = 4.5 nM T09572 C5SV9H 57396295 IC50 > 1000 nM T09572 C5W2PA 57396309 IC50 > 1000 nM T09572 CWJ94D 57396310 IC50 = 77 nM T09572 C4VP7L 57397816 IC50 = 120 nM T09572 CFXQ13 57397817 IC50 = 14 nM T09572 CNG7U5 57397818 IC50 = 141 nM T09572 C4ULN0 57397819 IC50 = 6 nM T09572 CP9SC0 57397820 IC50 = 27 nM T09572 CW0DC8 57398087 IC50 = 20 nM T09572 C80BEV 57398088 IC50 = 2.8 nM T09572 CM17JZ 57398089 IC50 > 1000 nM T09572 C4HM7E 57398090 IC50 > 1000 nM T09572 CRVU80 57398576 IC50 = 1000 nM T09572 CY6X5S 57399486 IC50 = 15 nM T09572 CRX4D5 57399487 IC50 = 179 nM T09572 C6DY7F 57399740 IC50 = 3.9 nM T09572 C3LYG6 57399741 IC50 = 12 nM T09572 CO2I5T 57399742 IC50 = 62 nM T09572 C0QHE2 57400241 IC50 = 400 nM T09572 C8A1RB 57400242 IC50 > 20000 nM T09572 CJ58YB 57401248 IC50 = 170 nM T09572 C2PC7Q 57401249 IC50 = 20 nM T09572 C2EHU3 57401250 IC50 = 30 nM T09572 C8OAM4 57401251 IC50 = 96 nM T09572 CB0M3A 57401252 IC50 = 30 nM T09572 CEM23S 57401507 IC50 = 19 nM T09572 CF71QU 57401508 IC50 = 70 nM T09572 CF97AB 57401509 IC50 = 6.7 nM T09572 CFY5N4 57401510 IC50 = 8.1 nM T09572 CMVO87 57401511 IC50 > 1000 nM T09572 C8MR2T 57401531 IC50 = 280 nM T09572 C34RTG 57402044 IC50 = 100 nM T09572 CLDV18 57402045 IC50 = 1000 nM T09572 C1ZPE7 57402226 IC50 = 136 nM T09572 CQI16H 57402500 IC50 = 450 nM T09572 CJFE03 57402992 IC50 = 20 nM T09572 CA6O0N 57402993 IC50 = 26 nM T09572 CHIW16 57403264 IC50 = 900 nM T09572 CV8HP7 57403265 IC50 > 1000 nM T09572 CFW3Y9 57403266 IC50 > 1000 nM T09572 CI5D1U 57403267 IC50 > 1000 nM T09572 C9MZU0 57403281 IC50 > 1000 nM T09572 C6WPC8 57403783 IC50 = 180 nM T09572 C7XW5S 57403784 IC50 = 3 nM T09572 CGO38J 57403785 IC50 = 50 nM T09572 C1L8YD 57404359 IC50 = 140 nM T09572 C8SX7A 57404360 IC50 = 110 nM T09572 C0Q1OZ 57404374 IC50 = 440 nM T09572 CXL13R 57521366 IC50 = 5.3 nM T09572 CV9ZT0 57522468 IC50 = 1.9 nM T09572 CRM9Q6 57522701 IC50 = 7.8 nM T09572 C7MT4F 57522703 IC50 = 2 nM T09572 CXUY90 57522704 IC50 = 4.4 nM T09572 C4EUO7 57522816 IC50 = 2.5 nM T09572 C6ZEW3 57522945 IC50 = 3.4 nM T09572 C2J8QB 57522946 IC50 = 2.4 nM T09572 CA2Y5C 57522947 IC50 = 2 nM T09572 CY2GW3 57522948 IC50 = 12 nM T09572 CF9X1V 57522949 IC50 = 5.5 nM T09572 CTPD32 57522950 IC50 = 3.8 nM T09572 C2WD7Q 57523086 IC50 = 1.5 nM T09572 CR7KU6 57845728 IC50 = 10 nM T09572 CPZ0W6 57890345 IC50 = 1 nM T09572 CDU52G 57890370 IC50 = 3 nM T09572 CXBS52 58423512 Ki = 13 nM T09572 C1YJH4 58646147 IC50 = 3.4 nM T09572 C6F4PY 59135471 IC50 = 50 nM T09572 CW8E6V 59135474 EC50 = 30 nM T09572 CO6TL1 59135478 EC50 = 30 nM T09572 CMNY97 59135479 IC50 = 63 nM T09572 C7WM1C 59135482 IC50 = 5.9 nM T09572 C7H4EZ 59135485 IC50 = 560 nM T09572 C2TD0S 59135486 IC50 = 230 nM T09572 CU4Z5R 59135490 IC50 = 340 nM T09572 CG1QE0 59135492 EC50 = 53 nM T09572 CDX98T 59691557 IC50 = 38 nM T09572 CUAY97 59691584 IC50 = 634 nM T09572 CDB34N 59691661 IC50 = 899 nM T09572 CV8U3A 59691704 IC50 = 94 nM T09572 C1MVB2 59835725 IC50 = 8 nM T09572 CZ6EF7 59835728 IC50 = 5 nM T09572 CMG1L8 59835758 IC50 = 8 nM T09572 C4Y8OJ 59835766 IC50 = 35 nM T09572 CG7JS4 59835780 IC50 = 4 nM T09572 C6I5DJ 59835799 IC50 = 12 nM T09572 C65CNM 59835853 IC50 = 10 nM T09572 CY30SJ 59835871 IC50 = 10 nM T09572 CK52CM 59835874 IC50 = 17 nM T09572 C42PAO 59835879 IC50 = 4 nM T09572 C4K2AL 59835909 IC50 = 78 nM T09572 C7SFO5 60130264 IC50 = 1 nM T09572 CA41LH 60130278 IC50 = 2 nM T09572 CIX06K 60130301 IC50 = 10 nM T09572 CIU8R5 60130302 IC50 = 29 nM T09572 C8HYR7 60130337 IC50 = 6 nM T09572 C70YHU 60130349 IC50 = 68 nM T09572 CGF54X 60150483 IC50 = 16 nM T09572 C1XTB5 60168816 IC50 = 70 nM T09572 CK0BH9 60168817 IC50 = 410 nM T09572 CA84NS 60168818 IC50 = 80 nM T09572 C0SJI9 60168913 IC50 = 120 nM T09572 C65BWQ 60168914 IC50 = 720 nM T09572 CE4I2W 60168915 IC50 = 160 nM T09572 C2S9DZ 60168916 IC50 = 1910 nM T09572 CJE24S 60169097 IC50 = 40 nM T09572 CNC6K8 60169098 IC50 = 60 nM T09572 C4BEU6 60169181 IC50 = 100 nM T09572 CD04TV 60169182 IC50 = 60 nM T09572 C7ZS9G 60169184 IC50 = 50 nM T09572 CU3X8A 60169185 IC50 = 80 nM T09572 CM8N0C 60169263 IC50 = 50 nM T09572 CO23GN 66877080 IC50 = 470 nM T09572 CX5H4B 69603769 IC50 = 220 nM T09572 C5AMB2 70681113 IC50 = 7 nM T09572 C59GPT 70681114 IC50 = 160 nM T09572 CO9Z6H 70681115 IC50 = 215 nM T09572 C8BP2U 70681116 IC50 = 158 nM T09572 CV0B8H 70681117 IC50 = 350 nM T09572 C4E1OI 70681197 IC50 = 171 nM T09572 CDH5M3 70681198 IC50 = 142 nM T09572 C14POJ 70681213 IC50 = 15 nM T09572 CV0X2S 70681214 IC50 = 20 nM T09572 C71GOK 70681215 IC50 = 66 nM T09572 CUWS85 70681216 IC50 = 21 nM T09572 CEP43U 70681217 IC50 = 19 nM T09572 C5MZT4 70681299 Ki = 210.86 nM T09572 C7HO6W 70683237 IC50 = 270 nM T09572 CYS92Z 70683241 IC50 = 59 nM T09572 C7FGW6 70683286 IC50 = 116 nM T09572 CL8FX4 70683287 IC50 = 30 nM T09572 CPJN73 70683299 IC50 = 81 nM T09572 CY7LX9 70683300 IC50 = 94 nM T09572 C3NR1Z 70683781 IC50 = 40 nM T09572 CXL0Y8 70685336 IC50 = 96 nM T09572 C53CDS 70685337 IC50 = 9 nM T09572 C08BEC 70685338 IC50 = 15 nM T09572 CDEZ93 70685346 IC50 = 258 nM T09572 CV0WI4 70685347 IC50 = 150 nM T09572 CCXF74 70685395 IC50 = 340 nM T09572 C2WS0G 70685396 IC50 = 86 nM T09572 CHZ6Y4 70685397 IC50 = 270 nM T09572 CYR86Q 70685398 IC50 = 26 nM T09572 CLUJ28 70685407 IC50 = 16 nM T09572 CH9EK3 70685408 IC50 = 69 nM T09572 CZO15N 70685409 IC50 = 4 nM T09572 C3HM0V 70685410 IC50 = 18 nM T09572 CXPR84 70687361 IC50 = 4000 nM T09572 CCRF61 70687470 IC50 = 146 nM T09572 CC3YQ9 70687471 IC50 = 180 nM T09572 CL79FG 70687472 IC50 > 10000 nM T09572 CALE31 70687473 IC50 = 18 nM T09572 C0YZF1 70687477 IC50 = 4 nM T09572 CEZ95O 70687478 IC50 = 237 nM T09572 C3P8VA 70687479 IC50 = 100 nM T09572 CEF40L 70687536 IC50 = 208 nM T09572 CPHD56 70687537 IC50 = 196 nM T09572 C59DKB 70687538 IC50 = 32 nM T09572 COY81J 70687549 IC50 = 31 nM T09572 CT8A1Y 70687550 IC50 = 26 nM T09572 C5UI4H 70687551 IC50 = 31 nM T09572 CE8FW5 70687552 IC50 = 26 nM T09572 CE6M1I 70688018 IC50 = 10 nM T09572 CGX8O4 70689518 IC50 > 10000 nM T09572 CT6NC1 70689519 IC50 = 91 nM T09572 C7GY1R 70689520 IC50 = 116 nM T09572 C7HY1M 70689525 IC50 = 27 nM T09572 C8K6GH 70689526 IC50 = 156 nM T09572 C1O6EB 70689527 IC50 = 59 nM T09572 CVYC02 70689594 IC50 = 40 nM T09572 C5JZ0U 70689595 IC50 = 54 nM T09572 C39VHU 70689596 IC50 = 91 nM T09572 C6RD9J 70689612 IC50 = 11 nM T09572 CQA6H0 70691333 IC50 = 22 nM T09572 C4GOS0 70691526 IC50 > 3000 nM T09572 CHX2V3 70691648 IC50 = 690 nM T09572 CJ8C3H 70691649 IC50 = 115 nM T09572 CC1G3W 70691650 IC50 = 33 nM T09572 CJ7VK5 70691651 IC50 = 45 nM T09572 C6HPK5 70691652 IC50 = 15 nM T09572 CYJS32 70691653 IC50 = 7 nM T09572 C7NI4U 70691655 IC50 > 10000 nM T09572 C2BEO6 70691656 IC50 = 67 nM T09572 CJQA94 70691720 IC50 = 107 nM T09572 C27ECJ 70691721 IC50 = 62 nM T09572 C9N0ZJ 70691722 IC50 = 24 nM T09572 CB71AI 70691723 IC50 = 230 nM T09572 CDI17T 70691724 IC50 = 4125 nM T09572 CM1W5S 70691725 IC50 = 35 nM T09572 CD3N0U 70691736 IC50 = 10 nM T09572 C31VLM 70691737 IC50 = 225 nM T09572 CK03LJ 70691738 IC50 = 14 nM T09572 C8CL4G 70691739 IC50 = 56 nM T09572 C4PH6G 70693620 IC50 = 3800 nM T09572 C2EGO8 70693732 IC50 = 30 nM T09572 C9Y0GP 70693733 IC50 = 3 nM T09572 C50FLK 70693734 IC50 = 10 nM T09572 C94PEU 70693737 IC50 = 33 nM T09572 C7R6XS 70693792 IC50 = 73 nM T09572 C0MN5C 70693793 IC50 = 83 nM T09572 CKTG14 70693794 IC50 = 575 nM T09572 C7OWB6 70693795 IC50 = 1800 nM T09572 CS79JT 70693796 IC50 = 57 nM T09572 CYE09Q 70693807 IC50 = 13 nM T09572 CHT37L 70693808 IC50 = 27 nM T09572 CY48LR 70693809 IC50 = 45 nM T09572 CO4G8Z 70693810 IC50 = 31 nM T09572 CA9NO7 70695565 Ki = 21 nM T09572 CYP9F5 70695851 IC50 = 246 nM T09572 C0CZ8Y 70695852 IC50 = 7300 nM T09572 C0OYQ4 70695853 IC50 = 163 nM T09572 C20EKP 70695854 IC50 = 213 nM T09572 CZ92AV 70695855 IC50 = 23 nM T09572 CJ61GF 70695859 IC50 = 208 nM T09572 C5SK0T 70695860 IC50 = 636 nM T09572 C6RM8L 70695913 IC50 = 670 nM T09572 CM6JE8 70695914 IC50 = 201 nM T09572 CY17NO 70695915 IC50 = 220 nM T09572 C7CF9D 70695916 IC50 = 182 nM T09572 C35IPG 70695917 IC50 = 255 nM T09572 CIW1D8 70695918 IC50 = 23 nM T09572 C8UD2I 70695929 IC50 = 170 nM T09572 CG0D4A 70695930 IC50 = 112 nM T09572 CW71LQ 70696356 IC50 = 0.76 nM T09572 C87MGT 71226277 IC50 = 20 nM T09572 C4J8MI 71226400 IC50 = 20 nM T09572 C1WP5Y 71226964 IC50 = 16 nM T09572 C1B9KV 71227161 IC50 = 45 nM T09572 CI8E6U 71227163 IC50 = 20 nM T09572 C26UYS 71450863 Ki = 3.9 nM T09572 CAEM97 71450908 Ki = 1188 nM T09572 CFEI76 71660915 IC50 = 40 nM T09572 C9I3GO 71714121 Ki = 14 nM T09572 CB2S3Z 71716477 IC50 = 4130 nM T09572 CF18UN 71716478 IC50 = 1040 nM T09572 CB0O6P 71716479 IC50 = 510 nM T09572 C5P6AH 71716480 IC50 = 5650 nM T09572 C0WF7K 71717084 IC50 = 3100 nM T09572 C2TNF8 71717085 IC50 = 10000 nM T09572 C0IL4X 71717086 IC50 = 2780 nM T09572 CNWZ92 71717700 IC50 = 340 nM T09572 CCLZ30 71717701 IC50 = 10000 nM T09572 CSZU90 71718317 IC50 = 210 nM T09572 C4JFS2 71718318 IC50 = 130 nM T09572 CIK12B 71718319 IC50 = 440 nM T09572 CKQ23I 71718910 IC50 = 180 nM T09572 CZOR72 71718911 IC50 = 7110 nM T09572 CMP54N 71719522 IC50 = 320 nM T09572 CVE7I3 71719523 IC50 = 190 nM T09572 CE0IQ4 71719524 IC50 = 2000 nM T09572 CJ9SP8 71719526 IC50 = 90 nM T09572 CK21FD 71720118 IC50 = 300 nM T09572 C2IJ4F 71720119 IC50 = 540 nM T09572 C3OM4R 71720120 IC50 = 80 nM T09572 C7D6VL 71720121 IC50 = 2010 nM T09572 CR1CA7 71730269 IC50 = 8.7 nM T09572 CF14LT 71730661 IC50 = 24 nM T09572 C7LX2Q 71730663 IC50 = 16 nM T09572 C9SN7I 71731948 IC50 = 33 nM T09572 CS5PA1 71732078 IC50 = 17 nM T09572 C8VJ7O 73356649 IC50 = 230 nM T09572 C1Q2HP 76324350 Ki <= 1500 nM T09572 C6BEM8 86582974 IC50 = 35 nM T09572 C1LJW9 89689924 IC50 = 12 nM T09572 C7S8ON 89690124 IC50 = 72 nM T09572 CHP67R 89690222 IC50 > 1000 nM T09572 CX01FB 89690237 IC50 = 92 nM T09572 CD3RU2 89690239 IC50 = 410 nM T09572 CP4Z8K 89690292 IC50 = 240 nM T09572 C9KT2U 89690293 IC50 > 1000 nM T09572 CK6AR1 89690294 IC50 > 1000 nM T09572 CRQ1S5 89690318 IC50 = 42 nM T09572 C7Y3BZ 89690333 IC50 > 1000 nM T09572 C24NIJ 89690365 IC50 = 37 nM T09572 C4W0KZ 89690368 IC50 = 380 nM T09572 C6TG1E 89690379 IC50 = 47 nM T09572 CJ42SW 89690396 IC50 = 24 nM T09572 C8IZG5 89690573 IC50 = 120 nM T09572 CG9X7P 89690574 IC50 = 7.7 nM T09572 CSQ84D 89690600 IC50 = 78 nM T09572 CLPT46 89690607 IC50 = 25 nM T09572 CJ6V7S 89690622 IC50 = 95 nM T09572 CN8VQ4 89690864 IC50 = 35 nM T09572 C8KT3J 89690957 IC50 = 34 nM T09572 CLI0S8 89690968 IC50 > 1000 nM T09572 CG1LS2 89690973 IC50 = 160 nM T09572 CQ0YA2 89691019 IC50 = 76 nM T09572 CE04BI 89691032 IC50 = 45 nM T09572 C0AYJ8 89691044 IC50 = 17 nM T09572 CU1X2I 89691057 IC50 = 85 nM T09572 C20YIN 89691065 IC50 = 41 nM T09572 C0XB6N 89691096 IC50 = 16 nM T09572 CE9C1Y 89691111 IC50 > 1000 nM T09572 CQB43P 89691143 IC50 = 100 nM T09572 CENL63 89691144 IC50 = 73 nM T09572 CP3I8Z 89691162 IC50 = 28 nM T09572 CZ5M8J 89691193 IC50 = 240 nM T09572 CUF15D 89691216 IC50 = 600 nM T09572 CZV10H 89691247 IC50 = 37 nM T09572 C9OV4S 89691264 IC50 > 1000 nM T09572 CZSL41 89691284 IC50 = 90 nM T09572 C9J6WL 89691349 IC50 > 1000 nM T09572 CHAI64 89691416 IC50 = 44 nM T09572 CX90VG 89691439 IC50 = 26 nM T09572 C2ZY0O 89691440 IC50 = 150 nM T09572 CP93JH 89691535 IC50 = 34 nM T09572 C50ODP 89702205 IC50 > 1000 nM T09572 CXR3A4 89702226 IC50 = 24 nM T09572 C4B8VD 89702233 IC50 = 17 nM T09572 CD94UH 89702341 IC50 > 1000 nM T09572 C0GS9K 89702355 IC50 = 180 nM T09572 C70YGQ 89702382 IC50 > 1000 nM T09572 CQE21B 89702566 IC50 = 14 nM T09572 C7BNF2 89798657 IC50 = 10 nM T09572 CYW7P8 89798658 IC50 = 13 nM T09572 C6BID5 90469437 IC50 = 38 nM T09572 C2IN9R 90666094 IC50 = 15 nM T09572 C9R7TC 90666095 IC50 = 3 nM T09572 C0KWI9 90666096 IC50 = 0.9 nM T09572 CXM6Q2 90666097 IC50 = 8 nM T09572 CMU2J7 90666098 IC50 = 34 nM T09572 CS71ZE 90666251 IC50 = 1004 nM T09572 CKV42Z 90666252 IC50 = 172 nM T09572 CIA63Z 90666253 IC50 = 817 nM T09572 C8YHD2 90666254 IC50 = 271 nM T09572 C90CGQ 90666255 IC50 = 138 nM T09572 CC07QH 90666256 IC50 = 47 nM T09572 CMO4T3 90666257 IC50 = 259 nM T09572 CWM0V6 90666258 IC50 = 3250 nM T09572 CT53ER 90666259 IC50 = 184 nM T09572 C6H5CY 90666260 IC50 = 46 nM T09572 CI2AQ3 90666261 IC50 = 651 nM T09572 CR0NA6 90666262 IC50 = 11 nM T09572 C8B5IV 90666263 IC50 = 27 nM T09572 CX6ZO5 90666264 IC50 = 15 nM T09572 C7J1IK 90666265 IC50 = 14 nM T09572 CCX69F 90666266 IC50 = 12 nM T09572 C45NLU 90666267 IC50 = 96 nM T09572 CR9HQ7 91759552 IC50 = 70 nM T09572 CS5A8P 91759588 IC50 = 57 nM T09572 C8XFV3 101007561 IC50 = 5128.61 nM T09572 CJMR89 117798671 IC50 = 90 nM T09572 CO2L5Z 117798675 IC50 = 140 nM T09572 C48XKW 117798680 IC50 = 230 nM T09572 CYU6B5 117798688 IC50 = 210 nM T09572 CN84IO 117798692 IC50 = 170 nM T09572 C54ISX 117798744 IC50 = 31 nM T09572 CM3F4S 117798780 IC50 = 130 nM T09572 CI2K4J 117816748 IC50 = 74 nM T09572 CL1Z6U 117816753 IC50 = 110 nM T09572 C1A3HV 117816804 IC50 = 43 nM T09572 CIET51 121386280 IC50 > 1000 nM T09572 C09BDS 122184557 IC50 = 2 nM T09572 CK35BS 122184558 IC50 = 8 nM T09572 CED1I6 122184559 IC50 = 470 nM T09572 C6JG4U 122184560 IC50 = 8 nM T09572 CTJO50 122184561 IC50 = 3 nM T09572 CZ1MA3 122184562 IC50 = 11 nM T09572 CH37IW 122184563 IC50 = 5 nM T09572 C5JTD9 122184564 IC50 = 36 nM T09572 CF2YG3 122184565 IC50 = 15 nM T09572 CRPW64 122184566 IC50 = 33 nM T09572 CACV74 122184567 IC50 = 700 nM T09572 CMR65S 122184568 IC50 = 420 nM T09572 CNC14U 122184569 IC50 = 360 nM T09572 CFC4P3 122184570 IC50 = 247 nM T09572 CJR48E 122184670 IC50 = 17 nM T09572 C7YA0Q 122184671 IC50 = 4 nM T09572 C6RP0N 122184672 IC50 = 21 nM T09572 CLP36J 122184673 IC50 = 151 nM T09572 CQT2K8 122184674 IC50 = 2530 nM T09572 CSIL49 122184687 IC50 = 251 nM T09572 CN0CB1 122184690 IC50 > 3000 nM T09572 C5Y0KX 122184691 IC50 = 95 nM T09572 C18ZKO 122184692 IC50 = 20 nM T09572 C0XJK1 122184693 IC50 = 6 nM T09572 C97APV 122184694 IC50 = 10 nM T09572 CLK94O 122184695 IC50 = 3 nM T09572 CWSF63 122184696 IC50 = 24 nM T09572 CW8L5K 122184697 IC50 = 9 nM T09572 CI4SF6 122184698 IC50 = 15 nM T09572 CDHE98 122184699 IC50 = 4 nM T09572 CIU9W5 122184700 IC50 = 92 nM T09572 CU2PG6 122184701 IC50 = 13 nM T09572 CKG74I 122184702 IC50 = 13 nM T09572 CZ0I1K 122184703 IC50 = 186 nM T09572 C65COE 122184704 IC50 = 15 nM T09572 CHS9N7 122184705 IC50 = 22 nM T09572 CWM9Q7 122184706 IC50 = 10 nM T09572 CZ2VB1 122184832 IC50 = 7 nM T09572 CJ0V1K 122184885 IC50 = 25 nM T09572 C2CHR3 123471111 IC50 = 34 nM T09572 CY6WF8 127025096 IC50 = 210 nM T09572 CELT51 127025110 IC50 = 270 nM T09572 C5IK3Q 127025395 IC50 = 94 nM T09572 CG28ML 127028868 IC50 = 69 nM T09572 CYP9E6 127028869 IC50 = 99 nM T09572 CS9YL7 127029623 IC50 = 3.8 nM T09572 CJO31V 127029624 IC50 = 3 nM T09572 C5P9RC 127029625 IC50 > 1000 nM T09572 C34PRW 127029630 IC50 > 1000 nM T09572 CK18EL 127029631 IC50 > 1000 nM T09572 C7S2DW 127029632 IC50 = 990 nM T09572 CFN3Y4 127029759 IC50 = 150 nM T09572 CZDO76 127030069 IC50 = 22 nM T09572 C8WD7N 127030070 IC50 = 23 nM T09572 C9GHX6 127030071 IC50 = 39 nM T09572 C0OKZ3 127030367 IC50 = 30 nM T09572 CEP0T2 127030368 IC50 = 35 nM T09572 CF4V0J 127031338 IC50 = 11 nM T09572 CZ6A2D 127031339 IC50 = 43 nM T09572 CZ6P7H 127031354 IC50 = 40 nM T09572 C5BTJ9 127031355 IC50 = 50 nM T09572 CB7XP0 127031356 IC50 = 39 nM T09572 C4F3QY 127031621 IC50 = 28 nM T09572 CB7Y6D 127031622 IC50 = 15 nM T09572 CUO4V9 127031623 IC50 = 44 nM T09572 CFG8U2 127031907 IC50 = 1000 nM T09572 CI9ZB4 127031908 IC50 = 61 nM T09572 C3NE8G 127031909 IC50 = 150 nM T09572 CYZH79 127032787 IC50 = 1200 nM T09572 C7AK5Z 127033095 IC50 = 75 nM T09572 C3UKI0 127033096 IC50 = 200 nM T09572 C9MD2C 127033672 IC50 = 140 nM T09572 C1YR3E 127033673 IC50 = 220 nM T09572 C5ITG3 127033945 IC50 = 70 nM T09572 C05XCQ 137635978 IC50 = 3235.94 nM T09572 C5PV0E 137640352 Ki = 15 nM T09572 CK5HG6 137644041 EC50 = 1042 nM T09572 CXH16S 137655884 IC50 = 1862.09 nM T09572 CME6U8 137657882 IC50 = 4265.8 nM T09572 CFC7Z0 155516078 IC50 = 17380 nM T09572 CX1A0M 155516949 IC50 = 6.8 nM T09572 C4TY3K 155520135 IC50 = 890 nM T09572 CLJU26 155522708 IC50 = 5100 nM T09572 CG4YE1 155524512 IC50 = 4300 nM T09572 CQ9PM4 155527803 IC50 = 129 nM T09572 C4AJ7V 155528494 IC50 = 105 nM T09572 C9RUQ4 155531314 IC50 = 4.9 nM T09572 CJ2S8K 155538229 IC50 = 40 nM T09572 CRC90P 155541584 IC50 > 3000 nM T09572 C0E4VQ 155562407 IC50 = 228 nM T09572 C6CTA5 155569743 IC50 = 1300 nM T09572 D00AWM 9826520 IC50 = 0.5012 nM T09572 D00MSU 22254580 IC50 = 492 nM T09572 D01NOZ 16665072 IC50 = 28 nM T09572 D01OYC 10262766 IC50 = 5310 nM T09572 D01OZL 10466405 IC50 = 36 nM T09572 D01PFN 22254575 IC50 = 432 nM T09572 D02FQG 54579974 IC50 = 25 nM T09572 D02QXF 11776033 IC50 = 860 nM T09572 D03BIQ 11189610 IC50 = 100 nM T09572 D03CDM 10399674 IC50 = 1070 nM T09572 D03FJK 10083869 IC50 = 20 nM T09572 D03FNQ 11281523 IC50 = 9 nM T09572 D03SEC 10443307 IC50 = 789 nM T09572 D04OOK 3787955 Ki = 7500 nM T09572 D05HFC 10466406 IC50 = 199 nM T09572 D05MEW 14514271 Ki = 302 nM T09572 D05QTT 11691555 Ki = 8.5 nM T09572 D05TVU 22254551 IC50 = 90 nM T09572 D05UZY 11539096 IC50 = 3 nM T09572 D05ZUX 44207909 EC50 = 128.82 nM T09572 D06KLQ 44403742 IC50 = 16 nM T09572 D07EPU 11155432 IC50 = 164 nM T09572 D07HQP 10353806 IC50 = 580 nM T09572 D07IUE 22254582 IC50 = 53 nM T09572 D07WFH 3575822 Ki = 7500 nM T09572 D07XEA 10332650 IC50 = 137 nM T09572 D08OQO 10198125 IC50 = 437 nM T09572 D08SOE 11994411 IC50 = 0.39 nM T09572 D09RGM 3747253 Ki = 1700 nM T09572 D0AT3U 44418001 IC50 = 1000 nM T09572 D0AT5N 56835134 IC50 = 1 nM T09572 D0AU6T 10377914 IC50 = 132 nM T09572 D0C5RQ 10300618 Ki = 19.95 nM T09572 D0C7ED 57523087 IC50 = 1.5 nM T09572 D0C9DP 11153928 IC50 = 9 nM T09572 D0D2PL 22266820 IC50 = 1590 nM T09572 D0ES2Y 22254604 IC50 = 32 nM T09572 D0F3VX 10466478 IC50 = 606 nM T09572 D0G6DS 10421932 IC50 = 818 nM T09572 D0I7FK 10038053 IC50 = 640 nM T09572 D0J7MM 11440762 IC50 = 390 nM T09572 D0K0KR 9895867 IC50 = 160 nM T09572 D0K5JA 10399494 IC50 = 361 nM T09572 D0K5QJ 11188955 IC50 = 70 nM T09572 D0K5XL 11440885 IC50 = 1930 nM T09572 D0L4WB 10244148 IC50 = 349 nM T09572 D0LJ4Q 10420382 IC50 = 1100 nM T09572 D0M3HZ 9927967 IC50 = 15 nM T09572 D0N6OL 11452268 IC50 = 58 nM T09572 D0P4CQ 10377822 IC50 = 191 nM T09572 D0P5QW 57521365 IC50 = 1.1 nM T09572 D0S7IJ 10083101 IC50 = 823 nM T09572 D0U1OX 10421933 IC50 = 201 nM T09572 D0V2IR 10353807 IC50 = 326 nM T09572 D0V9KF 22254540 IC50 = 722 nM T09572 D0W7ZM 10443853 IC50 = 614 nM T95558 D0EY0A 42636350 IC50 = 80 nM T95558 D02NRD 9865421 IC50 > 10000 nM T95558 D0M0NT 46926360 IC50 > 30000 nM T95558 D0U5NY 10435589 IC50 > 10000 nM T95558 CL21WZ 3168855 IC50 > 20000 nM T95558 C9A4YR 11892264 IC50 = 600 nM T95558 CKRN07 25118654 IC50 > 100000 nM T95558 CH3L6V 25192656 IC50 = 28000 nM T95558 C7URI3 25235407 IC50 > 10000 nM T95558 CM2G4X 42797508 IC50 > 50000 nM T95558 CAX57D 46850597 IC50 > 30000 nM T95558 CCY12P 46946735 IC50 > 50000 nM T95558 CW6EA0 52917768 IC50 = 1300 nM T95558 CBHT83 56840376 IC50 > 50000 nM T95558 CV8W4T 56933229 IC50 > 10000 nM T95558 C0QMK7 58064355 IC50 > 10000 nM T95558 C03EFU 59440893 IC50 > 30000 nM T95558 CW2LD6 70686525 IC50 > 20000 nM T95558 CY08FK 71571356 IC50 > 10000 nM T95558 C49QLP 71602372 IC50 > 10000 nM T95558 CR13XU 71602433 IC50 > 10000 nM T95558 C38SOR 71602434 IC50 > 10000 nM T95558 C3ZR8K 71603028 IC50 > 10000 nM T95558 CP97OC 71603093 IC50 > 10000 nM T95558 CAHY94 71603095 IC50 > 10000 nM T95558 C3IHF5 71603097 IC50 > 10000 nM T95558 CQ1K6W 71603210 IC50 > 10000 nM T95558 C9D1QC 71603211 IC50 > 10000 nM T95558 C8JKL2 71603212 IC50 > 10000 nM T95558 CJTR16 71766152 IC50 = 20 nM T95558 CVNX92 71766153 IC50 = 34 nM T95558 CGSV54 71766156 IC50 = 1.3 nM T95558 C5JV1P 71812623 IC50 > 20000 nM T95558 C9NE1Y 89853814 IC50 = 31 nM T95558 C47OKQ 89854212 IC50 = 17 nM T95558 C9FCS1 90644592 IC50 = 10000 nM T95558 CEC50G 91884614 IC50 > 30000 nM T95558 C4J9DB 118916617 IC50 = 120 nM T95558 C8EF1P 118916631 IC50 = 180 nM T95558 C2RBF7 118918048 IC50 = 2 nM T95558 CSBO65 122179027 IC50 > 30000 nM T95558 C75SHP 122188924 IC50 > 100000 nM T95558 C8HN7U 122189249 IC50 > 40000 nM T95558 CNV03S 122189255 IC50 > 100000 nM T95558 C48MIR 127034747 IC50 > 12000 nM T95558 C8UX4Q 127034759 IC50 = 540 nM T95558 CTM46H 127034938 IC50 = 500 nM T95558 C8VYP5 127034939 IC50 = 2200 nM T95558 C4OB5T 127035411 IC50 = 3 nM T95558 CUQ1Z6 127035947 IC50 = 140 nM T95558 CRI96L 127035948 IC50 = 1600 nM T95558 CTN0J4 127035949 IC50 = 300 nM T95558 CZV70W 127035950 IC50 = 60 nM T95558 CJ5OX8 127035951 IC50 = 3460 nM T95558 C1M5NI 127035952 IC50 = 4 nM T95558 CGET82 134586817 IC50 = 579 nM T95558 C6B5US 137628648 IC50 > 10000 nM T95558 C42PLT 145962320 IC50 > 50000 nM T95558 CLP89H 145963384 IC50 > 50000 nM T95558 C4MQU9 145980134 IC50 = 37 nM T95558 CQR0O2 155524798 IC50 = 17 nM T20302 D0ZD2M 16720766 IC50 > 1000 nM T20302 CP81AT 11655576 IC50 = 100000 nM T20302 C0YCU9 59671423 IC50 > 10000 nM T72702 D01FFA 72301 IC50 = 22.78 nM T72702 D0Y3KG 3121 IC50 = 1500000 nM T72702 D07SDQ 969516 IC50 = 13.16 nM T72702 D0I7IB 5222465 IC50 = 1000000 nM T72702 D0M8FD 4261 IC50 = 6000 nM T72702 C1WK2E 5417 IC50 = 14.98 nM T72702 CGO94B 34458 IC50 = 8.35 nM T72702 CQD56Z 73299 IC50 = 0.221 nM T72702 CEC2H3 73309 IC50 = 0.054 nM T72702 CHV19R 127026 IC50 = 6.46 nM T72702 C1ND9W 161665 IC50 = 152.43 nM T72702 C5Y6QK 261619 IC50 = 12.17 nM T72702 CHB7D2 453215 IC50 = 187.26 nM T72702 CS5PK2 640180 IC50 = 0.053 nM T72702 C2K4YZ 715840 IC50 = 13.37 nM T72702 CG1I7T 1550234 IC50 > 200 nM T72702 C4L7CX 1550330 IC50 = 0.26 nM T72702 CPU3R4 1550699 IC50 > 200 nM T72702 CC40IA 1909086 IC50 = 0.94 nM T72702 C5LGJ1 5282362 IC50 = 0.12 nM T72702 CM3T9J 5377817 IC50 = 15.39 nM T72702 C85WLD 5927890 IC50 = 141.98 nM T72702 CUYD15 9986341 IC50 = 0.095 nM T72702 CH5ZD8 10079039 IC50 = 9.581 nM T72702 CFJR86 11600024 IC50 = 36 nM T72702 C2VEB7 11753144 IC50 = 4.678 nM T72702 C56NRA 11957383 IC50 = 20 nM T72702 CF4W7L 12269810 IC50 = 968.9 nM T72702 CR0EG4 12302577 IC50 = 1.294 nM T72702 CCLH20 12313091 IC50 = 36.41 nM T72702 C4QK6B 13518132 IC50 = 15.95 nM T72702 C5U0AR 14189384 IC50 = 0.035 nM T72702 C6ZUG1 15061351 IC50 = 63.06 nM T72702 C5B1CH 15604798 Ki = 33 nM T72702 C6VZ1N 15942655 Ki = 800 nM T72702 CC5VF9 16007120 Ki = 2.6 nM T72702 CC7Y0D 16066741 IC50 = 590 nM T72702 CVB82P 17809181 IC50 = 89 nM T72702 C52BRP 21120798 IC50 = 0.28 nM T72702 CM87QX 21633122 IC50 = 10.61 nM T72702 CYE8Z0 23646853 Ki = 335 nM T72702 CF7JA3 23646854 Ki = 270 nM T72702 CRI3Y5 23646855 Ki = 350 nM T72702 CHUX39 23646856 Ki = 61.5 nM T72702 C6IT8J 23646857 Ki = 57 nM T72702 CFT69V 23646858 Ki = 130 nM T72702 C93HOM 23646859 Ki = 110 nM T72702 CTZ1K0 23646860 Ki = 100 nM T72702 CV3B5R 23646861 Ki = 330 nM T72702 CI2Q6A 23646862 Ki = 830 nM T72702 C2WK6E 23646863 Ki = 57 nM T72702 CVCZ14 23646864 Ki = 47 nM T72702 C2N6OU 23646865 Ki = 100 nM T72702 C6WGE2 23646866 Ki = 88 nM T72702 C54VSD 23646867 Ki = 28 nM T72702 C3GAY7 23646868 Ki = 60 nM T72702 CCD14G 23646869 Ki = 190 nM T72702 CXOF04 23646870 Ki = 58 nM T72702 C3W5LA 23646871 Ki = 160 nM T72702 CW5CX0 23646872 Ki = 130 nM T72702 CG91AX 23646873 Ki = 2700 nM T72702 CE75AW 23646874 Ki = 155 nM T72702 C4MO5W 23646875 Ki = 17000 nM T72702 CB8VS0 23646876 Ki = 130000 nM T72702 CU1L5O 23646877 Ki = 2000 nM T72702 C1COD6 23646878 Ki = 9500 nM T72702 CM5F3L 23646879 Ki = 220 nM T72702 CD01TF 23646880 Ki = 610 nM T72702 C58PMJ 23646881 Ki = 850 nM T72702 CXHL61 23646883 Ki = 72 nM T72702 C40ESI 44407593 IC50 = 120 nM T72702 CG3F5V 44407595 IC50 = 130 nM T72702 CJT68D 44407597 IC50 = 27 nM T72702 CH5L1B 44407599 IC50 = 31 nM T72702 C6M0JA 44407601 IC50 = 92 nM T72702 CLX0M1 44407607 IC50 = 210 nM T72702 CM8V2B 44407609 IC50 = 570 nM T72702 C4O0GT 44407611 IC50 = 180 nM T72702 CFZ12R 44407613 IC50 = 590 nM T72702 CMIF29 44407615 IC50 = 110 nM T72702 CX79CA 44407617 IC50 = 600 nM T72702 CCQ4O8 44407688 IC50 = 1600 nM T72702 C26PJY 44407814 IC50 = 47 nM T72702 C3GW8V 44407816 IC50 = 17 nM T72702 C7UCD4 44407818 IC50 = 150 nM T72702 C4S6FL 44407820 IC50 = 180 nM T72702 C51QCV 44407822 IC50 = 16 nM T72702 C5VW4Y 44407825 IC50 = 43 nM T72702 C2E0JC 44407841 IC50 = 48 nM T72702 C7QK8H 44407843 IC50 = 16 nM T72702 C36OIS 44407846 IC50 = 63 nM T72702 C3KTD2 44407848 IC50 = 170 nM T72702 CVSE54 44407974 IC50 = 240 nM T72702 C9N1SL 44407977 IC50 = 130 nM T72702 CW9L7N 44407979 IC50 = 2400 nM T72702 CUPX36 44407981 IC50 = 190 nM T72702 C71TKS 44407986 IC50 = 73 nM T72702 CGBR83 44407988 IC50 = 290 nM T72702 CZ69GQ 44408053 IC50 = 97 nM T72702 CJ3P4D 44408067 IC50 = 67 nM T72702 CG6H0U 44415561 Ki = 220 nM T72702 C3LCV6 44415581 Ki = 81 nM T72702 COY95B 44415713 Ki = 15 nM T72702 CSM18R 44415714 Ki = 20 nM T72702 CE3NH9 44415737 Ki = 1.3 nM T72702 CQ25XV 44421779 IC50 = 1300 nM T72702 CAP6F0 44421800 IC50 = 19000 nM T72702 CV1FC6 44421801 IC50 = 19000 nM T72702 CYE0W3 44421802 IC50 = 2200 nM T72702 CP1O3U 44421803 IC50 = 860 nM T72702 CNPU85 44421804 IC50 = 91000 nM T72702 CS3TC8 44421807 IC50 = 191000 nM T72702 C71ECV 44421808 IC50 = 8500 nM T72702 CF3AQ6 44421810 IC50 = 2400 nM T72702 CRX5K3 44421813 IC50 = 4200 nM T72702 C8OMB1 44421816 IC50 = 4200 nM T72702 C7VY0B 44421822 IC50 = 3200 nM T72702 CVJ85S 44421826 IC50 = 690 nM T72702 C4DYF3 44421831 IC50 = 300 nM T72702 CWVX31 44421837 IC50 = 150 nM T72702 CD58ZY 44421845 IC50 = 180 nM T72702 CQX8V2 44421851 IC50 = 300 nM T72702 CLV9Z6 46905970 IC50 = 380 nM T72702 CSX46R 57580978 IC50 = 376.52 nM T72702 C0B7OW 71508815 IC50 = 12.61 nM T72702 CA2LK1 71508816 IC50 = 118.8 nM T72702 C5GYN6 71508817 IC50 = 1501.43 nM T72702 CQDU73 71508864 IC50 = 555.37 nM T72702 CDB2C5 71508865 IC50 = 3.75 nM T72702 CQ2N0J 71508866 IC50 = 201.93 nM T72702 C2K3CV 71524613 IC50 = 6.75 nM T72702 C50YDS 71716758 IC50 = 38.59 nM T72702 CGU06V 71717958 IC50 = 8.79 nM T72702 CQY27U 71719784 IC50 = 16.8 nM T72702 CPK1H2 135450157 Ki = 2 nM T72702 CBU2E4 135469660 Ki = 44 nM T72702 CSW47P 135528873 Ki = 13 nM T72702 CQ3YN8 135530560 Ki = 4 nM T72702 C9Q7BK 135543038 Ki = 35 nM T72702 C9Q1TW 135543055 Ki = 43 nM T72702 C43KYW 135547926 Ki = 14 nM T72702 C89IBC 135547960 Ki = 13 nM T72702 CE2B7G 136094792 Ki = 12 nM T72702 CAW5Q0 136094793 Ki = 12 nM T72702 C2MZX6 137632271 IC50 = 0.028 nM T72702 C9HUM3 137634350 IC50 = 0.801 nM T72702 C61AWC 137635791 IC50 = 0.64 nM T72702 C3I4UR 137639091 IC50 = 0.078 nM T72702 CKNA04 137652993 IC50 = 0.221 nM T72702 D02KKU 12313704 IC50 = 0.221 nM T72702 D0IO0I 6474893 IC50 > 200 nM T72702 D0J6RQ 6437306 IC50 = 2.58 nM T72702 D0L7OM 6917970 IC50 = 104.58 nM T72702 D0PG8M 5467477 IC50 = 0.96 nM T72702 D0SJ2Q 10494 IC50 = 4.975 nM T72702 D0W1PV 6918328 IC50 = 200 nM T40103 D0J6AU 10152654 IC50 > 10 nM T40103 D0HM5J 118253852 IC50 > 20000 nM T40103 D04ZIJ 5478883 IC50 > 100000 nM T40103 CMW5A9 4430623 Ki = 251000 nM T40103 CESY50 5288259 IC50 > 500 nM T40103 C0XQP7 6917747 IC50 > 100000 nM T40103 CN26IL 9547980 Ki > 30000 nM T40103 COBW38 9821383 IC50 > 100000 nM T40103 CLB5G0 10025017 IC50 > 500 nM T40103 C2N9CS 10062713 IC50 = 18 nM T40103 CSO96K 10127748 IC50 > 5000 nM T40103 CKZ15P 10129236 IC50 > 5000 nM T40103 C5NEX6 10174161 IC50 > 5000 nM T40103 C1YR4T 10174359 IC50 > 2000 nM T40103 CY7DQ2 10288811 IC50 > 2000 nM T40103 CF5NB6 10668225 Ki = 160000 nM T40103 C5GD2S 10746284 Ki = 137000 nM T40103 CT9D8H 10765270 Ki = 210000 nM T40103 CG7D0X 10770036 Ki = 93000 nM T40103 CN0F8E 11199915 IC50 > 100000 nM T40103 CFI8L5 11502586 IC50 > 13000 nM T40103 C98EQF 11545899 IC50 = 230 nM T40103 CU57OC 11705307 IC50 > 100000 nM T40103 C8D7BS 11771234 Ki = 3700 nM T40103 CP4H9E 12737307 Ki = 89000 nM T40103 C31MCN 13186896 IC50 > 100000 nM T40103 C6XPN4 16664855 IC50 = 2653 nM T40103 CFY7O6 22988664 Ki = 354000 nM T40103 CZ8DI1 23643986 Ki = 137 nM T40103 CZPF48 23648277 IC50 > 50000 nM T40103 CN0VA7 24822701 IC50 > 50000 nM T40103 CQU38W 24900755 IC50 > 30000 nM T40103 C2S8VB 24901099 IC50 = 6591 nM T40103 CIN28B 24901100 IC50 > 10000 nM T40103 CD2EH0 24901101 IC50 > 10000 nM T40103 CS7B3F 24901102 IC50 > 100000 nM T40103 CGI0U2 25023791 Ki > 10000 nM T40103 C73KLE 25209862 IC50 > 30000 nM T40103 C25ELB 44143088 IC50 = 125.89 nM T40103 C9QDC0 44143091 IC50 = 645.65 nM T40103 C8Y9NQ 44219712 IC50 > 100000 nM T40103 C5VBI8 44368657 Ki = 260000 nM T40103 CP7KW2 44391459 IC50 = 580 nM T40103 C9W3HN 44391474 IC50 = 40 nM T40103 CV71WQ 44391475 IC50 = 8300 nM T40103 CTRP74 44394287 IC50 = 5000 nM T40103 CP7X6J 44394353 IC50 > 5000 nM T40103 C79NFU 44394458 IC50 > 12000 nM T40103 CD73QR 44398649 Ki = 0.46 nM T40103 CHQF16 44398651 Ki = 1.4 nM T40103 C4ALQ9 44398659 Ki > 13000 nM T40103 CD18YP 44402055 IC50 > 2000 nM T40103 CU8TB9 44402056 IC50 > 5000 nM T40103 CD4TP7 44402158 IC50 > 13000 nM T40103 CO6BG2 44402160 IC50 > 13000 nM T40103 C0AJC4 44402175 IC50 > 13000 nM T40103 CX9O2Q 44402263 IC50 > 13000 nM T40103 C89MOT 44402291 IC50 > 13000 nM T40103 C4ZMP9 44408016 IC50 > 13000 nM T40103 C25RIN 44408049 IC50 = 190 nM T40103 CS6X7V 44426055 IC50 > 100000 nM T40103 C8IB2W 44426056 IC50 > 100000 nM T40103 C8Z4WO 44459967 IC50 = 14454.4 nM T40103 C86ORE 44459987 IC50 = 16218.1 nM T40103 CLH74F 44565900 IC50 = 91760 nM T40103 CMIP10 44565901 IC50 > 100000 nM T40103 C70BXJ 44565925 IC50 = 66520 nM T40103 CS6YO0 44566187 IC50 = 145 nM T40103 CSF17Z 44566188 IC50 > 100000 nM T40103 CJP3U5 44566195 IC50 > 100000 nM T40103 CUFJ57 44566196 IC50 = 32570 nM T40103 CI7P2B 49797571 IC50 > 50000 nM T40103 CI59MV 49797572 IC50 > 50000 nM T40103 C96CKU 49797573 IC50 > 50000 nM T40103 CZM3L7 71520324 Ki = 129000 nM T40103 C63ROI 71717313 Ki = 221000 nM T40103 CGFK60 101201806 IC50 = 29000 nM T40103 C8E4WS 102323332 IC50 = 9800 nM T40103 C8X6JG 145970039 Ki = 329000 nM T40103 C51ZEH 145970706 Ki = 462000 nM T40103 CM53FT 145986712 Ki = 7000 nM T40103 CN6U8D 145988823 Ki = 108000 nM T40103 C5MWT1 145990477 Ki = 1300 nM T40103 CHD79T 44408017 IC50 > 13000 nM T40103 CO0N3S 44408050 IC50 > 13000 nM T40103 D05WZF 10129151 IC50 > 5000 nM T40103 D08KCA 72429 Ki = 9200 nM T40103 D09FGQ 123985 IC50 = 190 nM T40103 D0G2QG 44343301 IC50 = 40 nM T40103 D0L9VP 5287864 Ki = 1400 nM T40103 D0T7QF 10420833 IC50 > 13000 nM T40103 D0VE0F 10062714 IC50 > 13000 nM T40103 D0Y5IQ 44255320 IC50 = 10000 nM T34296 D00MDP 466151 Ki = 0.038 nM T34296 D04AIT 5280445 IC50 = 10050 nM T34296 D0K8KX 5280343 IC50 = 8460 nM T34296 D0S0LZ 54671203 IC50 = 40000 nM T34296 D05VZE 119031 IC50 = 2 nM T34296 D0A4RF 657061 IC50 = 0.6 nM T34296 D0HG5M 11452716 IC50 = 8 nM T34296 D0MW3H 9824350 Ki = 0.53 nM T34296 D0G1LL 74221072 IC50 = 47000 nM T34296 D0N6ZA 74221131 IC50 > 100000 nM T34296 D0UM5R 74221070 IC50 = 4800 nM T34296 D00UCC 9827497 IC50 = 3.3 nM T34296 D01DVX 9847838 IC50 = 461 nM T34296 D03BOZ 3342298 IC50 = 0.01 nM T34296 D0N8NK 11641563 IC50 = 4.7 nM T34296 D0P8YC 5362422 IC50 = 5 nM T34296 D0Q1CD 6918336 Ki = 1470 nM T34296 D0T9HG 132519 IC50 = 5.2 nM T34296 CNA81R 1836 Ki = 65 nM T34296 CZ45IU 4219 IC50 = 6.4 nM T34296 CFY8Q2 4230 IC50 = 1.3 nM T34296 C7ROG5 177347 IC50 = 1570 nM T34296 CV60YH 445010 IC50 = 3 nM T34296 C4D7TS 448002 IC50 = 3 nM T34296 CZDY56 645394 IC50 = 9900 nM T34296 CU6X2H 647218 IC50 = 15300 nM T34296 CY58CV 651056 IC50 = 4700 nM T34296 C4UMB1 651101 IC50 = 9400 nM T34296 C78NPG 651441 IC50 = 2500 nM T34296 CA70CP 664499 IC50 = 4000 nM T34296 CS4O7K 685005 IC50 = 31000 nM T34296 CP1Q6R 703233 IC50 = 67000 nM T34296 C2OCU9 779459 IC50 > 1000000 nM T34296 CEBX21 1016400 IC50 = 7700 nM T34296 CXNA13 1201165 IC50 = 4700 nM T34296 CH82ZT 1201321 IC50 = 1590 nM T34296 CAM10Y 1204907 IC50 = 640 nM T34296 C9IFC6 1348435 IC50 = 22000 nM T34296 C7K3JR 1358229 IC50 = 5890 nM T34296 C6UZ1A 1383990 IC50 = 6970 nM T34296 CVA63S 1506964 IC50 = 900 nM T34296 C4X0MZ 1870548 IC50 = 12600 nM T34296 CZ9TI3 2053915 IC50 = 39810.72 nM T34296 CN9C8D 2140735 IC50 = 120000 nM T34296 CJ3EF9 2221136 IC50 = 3600 nM T34296 CN6E3U 2366268 IC50 = 1900 nM T34296 CSL5X7 2369069 IC50 = 8100 nM T34296 CJ1LK6 2568387 IC50 = 25118.86 nM T34296 C0I9ZT 2571427 IC50 = 8400 nM T34296 C65UHI 2966106 IC50 = 6800 nM T34296 COH0C4 2994402 IC50 > 100000 nM T34296 C5Z9PF 2999799 IC50 = 13300 nM T34296 CO1HF6 3109990 IC50 = 24700 nM T34296 CP09YC 3109994 IC50 = 10900 nM T34296 CM72OK 3236108 IC50 = 12000 nM T34296 C5QT9A 3240046 IC50 = 3500 nM T34296 C6C3QR 3243814 IC50 = 23300 nM T34296 C0PB5H 3380837 IC50 = 177000 nM T34296 CME24U 3649035 IC50 = 24000 nM T34296 CT8PU3 3671894 IC50 > 67000 nM T34296 C3EI6T 4085085 IC50 = 14000 nM T34296 CBN96T 4358655 IC50 = 10000 nM T34296 CP8D7Y 4478236 IC50 = 75.86 nM T34296 CQ4VL5 5287415 IC50 = 0.7 nM T34296 CW5SE3 5288615 IC50 = 2.4 nM T34296 CJ3QI1 5288814 IC50 = 2330 nM T34296 C1R5CO 5289109 IC50 = 72 nM T34296 CA5D1J 5289110 IC50 = 8 nM T34296 CKM71T 5289111 IC50 = 6600 nM T34296 C7BPU5 5310930 IC50 > 40000 nM T34296 CVLS16 5319161 IC50 = 7620 nM T34296 C1CM3J 6005649 IC50 = 55270 nM T34296 C9S1VI 6006930 IC50 = 3990 nM T34296 C5OMB7 6102708 IC50 = 8 nM T34296 C0M3LR 6323382 IC50 = 3 nM T34296 CJG2B7 6476333 IC50 = 11090 nM T34296 CL5DH0 6479915 IC50 = 29030 nM T34296 CI86PQ 6539651 IC50 = 1.7 nM T34296 CQEF36 6539670 IC50 = 2 nM T34296 CP7BG0 6852146 IC50 = 1.3 nM T34296 CN5L2B 6852147 IC50 = 2.6 nM T34296 CP2XK7 6882342 IC50 = 140000 nM T34296 C0FQW9 7063077 Ki = 175 nM T34296 C9UPD8 9794928 IC50 = 1480 nM T34296 CA0ZH1 9798114 IC50 = 86 nM T34296 C7NP9Z 9798247 IC50 = 3 nM T34296 C78EKW 9798637 IC50 = 8 nM T34296 C80WFI 9800763 IC50 = 4.4 nM T34296 C76RCQ 9801569 IC50 = 155 nM T34296 C68HMJ 9801786 IC50 = 3019.95 nM T34296 CM9GH8 9802180 IC50 = 1 nM T34296 CIXD67 9802768 IC50 < 1 nM T34296 C83FVW 9803207 IC50 = 1 nM T34296 C3QS5H 9803407 IC50 = 47 nM T34296 CUSD58 9803469 IC50 = 89 nM T34296 C4QCG9 9803771 IC50 = 5 nM T34296 C23VTC 9804342 IC50 = 3 nM T34296 C49HNU 9805016 IC50 = 1 nM T34296 CXSU10 9805304 IC50 = 83 nM T34296 CO4D0U 9805473 IC50 = 1 nM T34296 C1HP7E 9805710 IC50 = 67 nM T34296 CT8X1F 9806970 IC50 = 321 nM T34296 CTK6J8 9808181 IC50 = 2300 nM T34296 C67XKV 9808391 IC50 = 3 nM T34296 CS07BM 9808594 IC50 = 3 nM T34296 C9RQM7 9808674 IC50 = 0.35 nM T34296 C5CE8A 9809470 IC50 = 4.5 nM T34296 C32ODL 9818295 IC50 = 182 nM T34296 C0R2KN 9818588 IC50 > 10000 nM T34296 CC9VY4 9819420 IC50 = 33 nM T34296 C1VT4J 9819974 IC50 = 26 nM T34296 CQG86S 9820708 IC50 = 2 nM T34296 CN4AP6 9821427 IC50 = 3.49 nM T34296 C6KJ9W 9822461 IC50 = 5.3 nM T34296 C6IX7G 9822926 IC50 = 0.15 nM T34296 CVN5Z3 9823395 IC50 = 30 nM T34296 CUZ25T 9825237 IC50 = 9 nM T34296 C3AEF4 9825692 IC50 = 5 nM T34296 CDJB86 9825720 IC50 = 0.016 nM T34296 CXL65P 9825920 Ki > 5000 nM T34296 CL0G8K 9825927 IC50 = 100 nM T34296 CVSJ72 9826275 IC50 = 1 nM T34296 C7W3TG 9826481 IC50 = 289 nM T34296 CPW60S 9827023 IC50 = 34.6 nM T34296 CXTY18 9827218 IC50 = 290 nM T34296 C24CZI 9827635 IC50 = 7 nM T34296 C2TU0C 9827807 IC50 = 2 nM T34296 CC1NG5 9829581 IC50 = 20 nM T34296 C8WH1Q 9840355 IC50 = 14 nM T34296 CU7FM2 9840390 IC50 = 44 nM T34296 CEAZ87 9840395 IC50 = 84 nM T34296 C9PW7L 9841168 Ki = 206 nM T34296 C5XL7R 9841323 IC50 = 0.2 nM T34296 CRP01H 9841401 Ki = 130 nM T34296 CA7DJ9 9842114 IC50 = 2.4 nM T34296 CQ5L0D 9842167 IC50 = 500 nM T34296 CH63ZI 9842332 IC50 = 12 nM T34296 CC1TB5 9842343 IC50 = 148 nM T34296 C6YT5W 9843479 IC50 = 41.5 nM T34296 C9N5PA 9843679 IC50 = 0.77 nM T34296 C49UOA 9844245 IC50 = 6.5 nM T34296 CK76RW 9845271 IC50 = 29 nM T34296 CD31XZ 9845513 IC50 = 365 nM T34296 CEB90C 9846418 IC50 = 1 nM T34296 C4D2MY 9846507 IC50 = 2 nM T34296 C0KP9H 9847092 IC50 = 2 nM T34296 CE9AL3 9847113 IC50 < 0.1 nM T34296 C6SV1X 9847843 IC50 = 1 nM T34296 CG14CO 9848625 IC50 = 358 nM T34296 C92EJW 9849379 IC50 = 5 nM T34296 CX3EW2 9849576 IC50 = 155 nM T34296 CHVL24 9849957 IC50 = 3 nM T34296 C4IEK0 9850035 IC50 = 0.2 nM T34296 C9P1BH 9851086 IC50 = 1 nM T34296 C5DGI9 9851911 IC50 = 4.5 nM T34296 CC70WV 9858468 IC50 = 107 nM T34296 CECR39 9860227 IC50 = 3450 nM T34296 CR37HQ 9861014 IC50 = 751 nM T34296 C5TUJ7 9862317 IC50 = 7 nM T34296 CS5JT6 9864502 IC50 = 4 nM T34296 CGUF07 9865358 IC50 = 5.7 nM T34296 CU51IV 9865936 IC50 = 2 nM T34296 CI8Z0R 9866250 IC50 = 0.75 nM T34296 CP4Y7O 9867411 IC50 = 6 nM T34296 C0YN1X 9867935 IC50 = 33 nM T34296 CK3F1T 9868079 IC50 = 28 nM T34296 C2L9SU 9868329 IC50 = 2 nM T34296 CJS23I 9868333 Ki > 5025 nM T34296 C5O0GC 9868490 IC50 = 97 nM T34296 CRI23M 9868515 IC50 = 52 nM T34296 C4K2GH 9868577 IC50 = 2 nM T34296 C4ZR7O 9868713 IC50 = 77 nM T34296 C24JSB 9868858 IC50 = 33 nM T34296 C5IJH2 9869068 IC50 = 15 nM T34296 CT76IN 9869441 IC50 = 2 nM T34296 CA6G0W 9869598 IC50 = 2 nM T34296 CZO6K4 9869819 IC50 = 0.4 nM T34296 C5ELS6 9869902 IC50 = 2 nM T34296 CMEA71 9869947 IC50 = 1.1 nM T34296 CA48SX 9870269 IC50 = 1.9 nM T34296 C25-SEP 9870933 IC50 = 701 nM T34296 C5QFG1 9871290 IC50 = 2 nM T34296 CSM16R 9871355 IC50 = 302 nM T34296 CHU9I8 9871883 IC50 = 0.1 nM T34296 CU9L3X 9879183 IC50 > 10000 nM T34296 CG41SV 9879575 IC50 > 10000 nM T34296 C0TCJ2 9880675 Ki = 904 nM T34296 C0NA6S 9880842 IC50 = 100 nM T34296 C0QY4U 9883809 IC50 = 946 nM T34296 C9XSN0 9883962 IC50 = 4760 nM T34296 C2OHV3 9885051 IC50 = 34 nM T34296 CKFD90 9885716 IC50 = 38 nM T34296 CG35XZ 9885916 IC50 = 1000 nM T34296 CZBK85 9886177 IC50 = 78 nM T34296 CHT08B 9886916 IC50 = 0.65 nM T34296 C2M4EC 9887473 Ki > 5025 nM T34296 C1STP9 9887771 IC50 = 1.2 nM T34296 CFG4Q2 9887831 IC50 = 9 nM T34296 C3ZG6O 9887870 IC50 = 8 nM T34296 CC87LP 9888280 IC50 = 2 nM T34296 CD76WB 9888485 IC50 = 2 nM T34296 CVP45O 9888530 IC50 = 231 nM T34296 CJS0E5 9888649 IC50 = 8 nM T34296 CB2YG7 9889128 IC50 = 2 nM T34296 CD1U5P 9889190 IC50 = 20.89 nM T34296 C4AVN6 9889449 IC50 = 200 nM T34296 CZD2E3 9889870 IC50 = 4 nM T34296 C26SZX 9890226 IC50 = 0.6 nM T34296 CWN19T 9890526 IC50 = 12.2 nM T34296 CD79UJ 9890632 IC50 > 100000 nM T34296 CNX78A 9890733 IC50 = 1 nM T34296 CMD0S2 9891009 IC50 = 47 nM T34296 C20LGF 9891255 IC50 = 31 nM T34296 C9YD2O 9891259 IC50 = 16 nM T34296 CU65HY 9891358 IC50 = 1.2 nM T34296 C3QSE6 9891814 IC50 = 5 nM T34296 CPT4C6 9892042 IC50 = 427 nM T34296 CR50BS 9892336 IC50 = 27 nM T34296 C1KV7J 9892518 IC50 = 26 nM T34296 CH69LT 9892815 IC50 < 0.1 nM T34296 CZU7Y4 9892876 IC50 = 129 nM T34296 CX82KN 9893236 IC50 = 1.4 nM T34296 C2G5AQ 9894201 IC50 = 908 nM T34296 CSIB97 9896504 IC50 = 23 nM T34296 C6Q4JF 9903007 IC50 = 22 nM T34296 C2R5CX 9905493 IC50 = 1.8 nM T34296 CD78ZQ 9907286 IC50 = 0.9 nM T34296 CYHN04 9908006 IC50 = 7 nM T34296 CKWF30 9908681 IC50 = 22 nM T34296 CQ8Y9T 9909624 IC50 = 0.37 nM T34296 CJ3K1I 9910075 IC50 = 2137.96 nM T34296 C4E6LR 9910544 IC50 = 150 nM T34296 C6NUE9 9910550 IC50 = 3 nM T34296 CP4LS8 9910727 IC50 = 498 nM T34296 C2GMQ0 9912235 IC50 = 119 nM T34296 C62VZI 9912382 IC50 = 12 nM T34296 C8VJ9Z 9913053 IC50 = 1 nM T34296 CI5A3G 9913301 IC50 = 3 nM T34296 C3AZP0 9913479 IC50 = 1.4 nM T34296 CX1Q5C 9913489 IC50 = 1 nM T34296 C7ZY1L 9914029 IC50 = 248 nM T34296 CU9B3E 9914147 IC50 = 20 nM T34296 CX3C2G 9914326 IC50 = 72 nM T34296 CM39FU 9915194 IC50 = 2377 nM T34296 CA3FW0 9918908 IC50 = 0.008 nM T34296 CM7UO8 9924798 IC50 = 24 nM T34296 CBPD13 9926779 IC50 = 37 nM T34296 CSA12Z 9927353 IC50 = 57 nM T34296 C26ZPC 9929976 IC50 = 2 nM T34296 C1KX3E 9930058 IC50 = 2 nM T34296 CLJ61Q 9931505 IC50 = 2 nM T34296 C67PBX 9932128 IC50 = 11 nM T34296 CJI5A7 9932167 IC50 = 2 nM T34296 CY79AT 9932263 IC50 = 1.2 nM T34296 C03GVA 9932290 Ki = 210 nM T34296 C3VO2E 9932958 IC50 = 12 nM T34296 CT2KM9 9933083 IC50 = 100 nM T34296 CDXR37 9933197 IC50 = 0.4 nM T34296 C2EUL8 9933259 IC50 = 34 nM T34296 CX17KQ 9933408 IC50 = 104.71 nM T34296 C57WSD 9934240 IC50 = 42 nM T34296 CGJZ78 9934997 IC50 = 29 nM T34296 C65ION 9935032 IC50 = 0.2 nM T34296 C1HRU9 9936228 IC50 = 3.8 nM T34296 CDRC76 9936405 IC50 = 317 nM T34296 CH9G5D 9936469 IC50 = 9.5 nM T34296 C7GJF8 9936712 IC50 = 5 nM T34296 CG38KL 9936728 Ki = 2.3 nM T34296 CE59TP 9936926 IC50 = 758.58 nM T34296 C12ZGS 9945200 IC50 = 396 nM T34296 C0MLZ6 9945553 IC50 = 2000 nM T34296 CA30JY 9946988 IC50 = 520 nM T34296 C6TH4I 9947270 IC50 = 708 nM T34296 C16HTN 9948666 Ki = 17 nM T34296 C52IUJ 9949603 IC50 = 2000 nM T34296 CWO48K 9952436 IC50 = 1.5 nM T34296 C8C3DL 9953278 IC50 = 580 nM T34296 C9OY4Z 9953817 IC50 = 9 nM T34296 CABI45 9954117 IC50 = 11 nM T34296 C8RXN6 9954304 IC50 = 869 nM T34296 C6GA8D 9954513 IC50 = 11 nM T34296 CH9YL3 9954604 IC50 = 3 nM T34296 C37VXK 9954605 IC50 = 2 nM T34296 CK9HX0 9955125 IC50 = 0.4 nM T34296 CMV37W 9955127 IC50 = 49 nM T34296 CWE6N8 9955640 IC50 = 3 nM T34296 C3ZLA1 9956465 IC50 = 40 nM T34296 C3Q2UJ 9956686 IC50 = 0.25 nM T34296 C56GFP 9956833 IC50 = 3 nM T34296 CQ80MP 9957107 IC50 = 7 nM T34296 C5I0VJ 9957500 IC50 = 233 nM T34296 CN76XI 9957653 IC50 = 1 nM T34296 CPJR82 9957875 IC50 = 3 nM T34296 CYJ35F 9958085 IC50 = 0.12 nM T34296 CWE4D3 9958604 IC50 = 6 nM T34296 CNHT34 9959421 IC50 = 0.4 nM T34296 CN8TK0 9959428 IC50 = 1691 nM T34296 C9DRB7 9966028 IC50 = 185 nM T34296 CYK75X 9967932 IC50 > 10000 nM T34296 C0HL2X 9976697 IC50 = 0.9 nM T34296 C09LSY 9979489 Ki > 5025 nM T34296 CUA65C 9982414 IC50 = 0.95 nM T34296 CO09PN 9983251 IC50 = 0.9 nM T34296 CJGR30 9983604 IC50 = 0.7 nM T34296 C3KX1B 9998685 Ki = 3 nM T34296 C8W5UK 9999879 IC50 = 527 nM T34296 C59WEK 10001843 IC50 < 0.1 nM T34296 CR7T3J 10009978 Ki = 50 nM T34296 CJ6H8O 10019658 IC50 = 1 nM T34296 C71YGT 10025307 Ki = 4.169 nM T34296 C5PKZ1 10029419 IC50 = 0.09 nM T34296 CM52RO 10030422 IC50 = 14 nM T34296 CJR59P 10031295 Ki > 5025 nM T34296 C7J9ZF 10039403 IC50 = 64 nM T34296 CNA3G4 10042214 IC50 = 12 nM T34296 C07DLO 10046817 IC50 = 290 nM T34296 CHF92V 10047100 Ki = 2.692 nM T34296 CLXN48 10047373 IC50 = 1 nM T34296 C1N9UX 10050222 IC50 = 154 nM T34296 CLZ87W 10051236 Ki = 753 nM T34296 C21ULC 10052150 IC50 = 0.16 nM T34296 CSHD67 10054852 IC50 = 0.4 nM T34296 CJK0R1 10074190 IC50 = 1 nM T34296 CPS4R9 10076090 IC50 = 0.8 nM T34296 CPKC43 10093147 IC50 = 4 nM T34296 C5W4ZA 10094362 IC50 = 40 nM T34296 C2XV5J 10098250 IC50 = 1 nM T34296 C3V2HW 10099112 IC50 = 12 nM T34296 CXV2Y3 10109170 Ki = 1055 nM T34296 C0G7IY 10114318 Ki = 470 nM T34296 C9T2AW 10116042 IC50 = 10 nM T34296 CVK61T 10116047 IC50 = 11 nM T34296 C78JHL 10116107 Ki = 570 nM T34296 CP5L0W 10117663 Ki = 3869 nM T34296 C7OPQ8 10118047 IC50 = 0.4 nM T34296 CU3ZM2 10118633 IC50 > 1000 nM T34296 C2F8KW 10119294 IC50 = 1 nM T34296 CPA4R9 10119730 IC50 = 7 nM T34296 C7A8MI 10120093 IC50 = 0.2 nM T34296 C0Q9DW 10120586 IC50 = 20 nM T34296 C0KHW5 10120930 IC50 = 50 nM T34296 CP65KL 10125869 Ki = 55 nM T34296 CPTG57 10126378 IC50 = 122 nM T34296 CY2N3D 10127629 Ki > 5020 nM T34296 C1N4MJ 10127670 Ki > 5020 nM T34296 CIL09Z 10127889 Ki > 5020 nM T34296 CYU19P 10127901 Ki = 3530 nM T34296 C07KFI 10128313 Ki > 5020 nM T34296 CB3I6K 10128659 Ki > 5020 nM T34296 C6ZK3A 10128916 Ki > 5020 nM T34296 CS54CQ 10133565 IC50 > 10000 nM T34296 C0SVY1 10134897 IC50 = 4019 nM T34296 C9EWX5 10135125 IC50 = 13 nM T34296 C7KR3Y 10136680 Ki = 320 nM T34296 CNU93J 10136924 Ki = 650 nM T34296 C1CDF2 10136925 Ki = 300 nM T34296 CJ9EX4 10138303 Ki = 3810 nM T34296 C6UXD7 10138936 IC50 = 85 nM T34296 CU6Y9T 10140438 Ki > 5025 nM T34296 CE75BY 10140776 Ki = 1206 nM T34296 CIH36M 10141214 IC50 = 0.2 nM T34296 C5DA1U 10141270 IC50 = 4 nM T34296 C5H1ZM 10141426 IC50 = 1 nM T34296 C6MSI0 10141443 IC50 = 7300 nM T34296 CLXF15 10141613 Ki > 5000 nM T34296 C7VF1K 10141614 Ki = 2613 nM T34296 CWB5O4 10142326 Ki > 5000 nM T34296 CPXB21 10143028 Ki > 5025 nM T34296 C23WZR 10143587 Ki > 5000 nM T34296 CAM6U7 10143672 IC50 = 6 nM T34296 C82SMW 10144091 IC50 = 3 nM T34296 CD3U8E 10150649 Ki = 7 nM T34296 CJMV83 10152887 IC50 = 3.3 nM T34296 CZW98O 10156375 Ki = 55 nM T34296 CPY87U 10158366 IC50 > 10000 nM T34296 CYO8D2 10159633 Ki > 5025 nM T34296 CHUA34 10160545 IC50 = 2.4 nM T34296 CQ41YI 10161391 Ki > 5025 nM T34296 CCU9S1 10162155 IC50 = 1 nM T34296 C7SXD4 10162245 Ki = 3266 nM T34296 CO6PS3 10162900 Ki = 130 nM T34296 CR5H6E 10163627 Ki > 5025 nM T34296 CZO5V4 10164317 IC50 = 0.4 nM T34296 CCM0Y8 10165180 Ki = 603 nM T34296 CE10MK 10165419 IC50 = 7 nM T34296 CP02FJ 10165420 IC50 = 7 nM T34296 C0K7HT 10165868 IC50 = 1 nM T34296 C9X8YZ 10172500 IC50 = 130 nM T34296 CB3Q9L 10172753 IC50 = 61.2 nM T34296 CA81UR 10173271 IC50 = 10000 nM T34296 C6IW4O 10173876 Ki > 5020 nM T34296 CV7ES2 10174780 IC50 = 1.7 nM T34296 C8NAM9 10174791 IC50 = 1 nM T34296 CN6I1L 10174798 IC50 = 0.54 nM T34296 CZL72O 10175020 IC50 = 0.45 nM T34296 C4QY3V 10175210 Ki = 5020 nM T34296 C84ZQD 10175219 Ki = 1310 nM T34296 C5JM1A 10179045 IC50 > 10000 nM T34296 CD4AO0 10180362 IC50 = 2200 nM T34296 CCX3T6 10183064 Ki > 15000 nM T34296 CS6X2R 10183408 IC50 = 2 nM T34296 C6OE9H 10183692 IC50 > 10000 nM T34296 CDM94B 10183693 Ki > 5000 nM T34296 C2GV5Q 10183755 IC50 = 65 nM T34296 CH04IS 10184457 IC50 = 2 nM T34296 C3E9NF 10184537 Ki > 5000 nM T34296 CTDP62 10184579 Ki > 5000 nM T34296 CXQ8N0 10185100 Ki = 3136 nM T34296 C2OM9G 10186288 IC50 = 16 nM T34296 CK0P3F 10186536 Ki > 5025 nM T34296 CV7YI1 10186544 Ki > 5000 nM T34296 CA9FG4 10187181 IC50 = 4 nM T34296 CY9W6L 10194183 IC50 = 13.5 nM T34296 C51RPY 10195069 Ki > 5020 nM T34296 CY36NO 10196425 Ki > 5020 nM T34296 C63JGO 10196445 IC50 = 0.68 nM T34296 C0U9KC 10199401 IC50 = 32 nM T34296 C5CUM9 10202769 Ki > 5025 nM T34296 CX8BS3 10203685 Ki > 5025 nM T34296 C4FSU0 10203714 IC50 = 0.88 nM T34296 CE1LI3 10204303 Ki = 120 nM T34296 C32RAQ 10204620 Ki > 5000 nM T34296 C7AU0H 10205886 IC50 = 26 nM T34296 CQFP69 10206106 Ki = 370 nM T34296 CS1CA5 10207780 Ki = 653 nM T34296 C4K1MJ 10208262 Ki > 5025 nM T34296 CV4DG9 10209314 IC50 = 2 nM T34296 CD76KE 10209382 Ki > 5025 nM T34296 CT62UX 10215925 IC50 = 57 nM T34296 CVQA31 10216178 IC50 = 18 nM T34296 CXRT17 10218227 IC50 = 0.73 nM T34296 C7Y2US 10218353 Ki = 3720 nM T34296 C1C7AH 10223757 Ki > 5025 nM T34296 C92BVJ 10223963 IC50 = 21 nM T34296 CV5X8A 10224181 IC50 = 0.67 nM T34296 CGKU70 10224396 Ki = 250 nM T34296 C7K1OR 10224602 IC50 = 2000 nM T34296 CLH71C 10225319 Ki > 5025 nM T34296 C2X1KF 10226116 Ki = 753 nM T34296 C9CSG3 10226996 IC50 = 8.2 nM T34296 CJ46HR 10227522 IC50 = 2 nM T34296 CUE63Q 10227853 Ki > 5000 nM T34296 C19DFP 10227854 Ki > 5000 nM T34296 CSDG58 10228529 IC50 = 255 nM T34296 C7T0WH 10229644 IC50 = 1.8 nM T34296 CD2HP3 10230012 Ki > 5000 nM T34296 CLJ3Y9 10230286 IC50 = 1 nM T34296 CCRM18 10231253 IC50 = 1.1 nM T34296 CCTY95 10237492 Ki = 5020 nM T34296 CRF32B 10237550 Ki = 10 nM T34296 CNO8Z1 10237571 IC50 = 1.54 nM T34296 CF5PO0 10237938 IC50 = 3000 nM T34296 CWR7E2 10237960 IC50 = 6.5 nM T34296 CBG59O 10238145 IC50 = 13.9 nM T34296 C91DMB 10239619 IC50 = 0.36 nM T34296 CG70QJ 10239685 IC50 = 0.93 nM T34296 CCQ9V5 10239716 Ki > 5020 nM T34296 C8LQP4 10253358 IC50 = 0.65 nM T34296 C2V4MP 10253549 IC50 = 1.9 nM T34296 CQF3V9 10253673 IC50 = 34.67 nM T34296 CJKD83 10268288 IC50 > 10000 nM T34296 CMNA19 10270268 IC50 > 10000 nM T34296 C2MES9 10271604 Ki = 91000 nM T34296 CBJE75 10272162 IC50 = 11.7 nM T34296 CGP97S 10274748 Ki = 180 nM T34296 CU67RC 10275101 IC50 = 2.7 nM T34296 CES6A5 10276821 Ki = 804 nM T34296 C0GU6B 10277568 IC50 = 2 nM T34296 CY6K1G 10277706 Ki = 3266 nM T34296 C9OAE1 10277812 IC50 = 3 nM T34296 C2UAM8 10278729 IC50 = 1 nM T34296 C5Z2IG 10278742 IC50 = 0.8 nM T34296 C6KR5M 10278934 IC50 = 9 nM T34296 C3IG0K 10280852 IC50 < 0.1 nM T34296 C7TWG0 10289551 Ki > 5020 nM T34296 CJ63ER 10289607 Ki > 5020 nM T34296 CR48SA 10289842 Ki > 5210 nM T34296 CP0I5Y 10291146 IC50 > 10000 nM T34296 CLP72J 10293348 IC50 > 10000 nM T34296 CS69YG 10293394 IC50 = 9000 nM T34296 CB82ZF 10294766 IC50 = 90 nM T34296 CDU36Y 10296475 Ki = 1330 nM T34296 C48IRP 10296785 Ki = 140 nM T34296 CQ1Z0G 10298111 IC50 = 900 nM T34296 CN14MI 10298369 Ki > 5025 nM T34296 C25EKM 10299665 Ki = 753 nM T34296 C1BR6A 10300063 Ki > 5025 nM T34296 C80VEU 10300077 Ki > 5025 nM T34296 CFAU84 10301584 Ki > 5025 nM T34296 CP5AU1 10302088 Ki > 5025 nM T34296 C35LHB 10309800 IC50 = 244 nM T34296 CE1C7H 10310082 IC50 = 0.15 nM T34296 CE1KM9 10311498 Ki = 3950 nM T34296 C4MC8P 10311673 IC50 = 2 nM T34296 CP3D5K 10311698 IC50 = 0.57 nM T34296 COBH25 10311898 IC50 = 0.88 nM T34296 C4R9ZK 10311997 Ki = 95 nM T34296 CE6MB0 10312141 Ki = 356 nM T34296 CDO9J3 10318516 Ki = 110 nM T34296 CIDW49 10319098 Ki > 5025 nM T34296 CG23FV 10320328 IC50 = 0.6 nM T34296 CJ6XM1 10321516 IC50 = 1 nM T34296 CJWH74 10321975 Ki > 5025 nM T34296 CY08WJ 10322755 Ki > 5000 nM T34296 C3QDH0 10340642 Ki = 1.9 nM T34296 CL8YC0 10346590 IC50 = 0.05 nM T34296 C94ANQ 10347529 IC50 = 0.8 nM T34296 C4K9MO 10355923 Ki = 2200 nM T34296 CWIM61 10364088 IC50 = 10 nM T34296 CL4B2U 10364155 IC50 = 16900 nM T34296 CI0T8K 10366352 Ki > 5025 nM T34296 CBTO07 10370226 Ki > 5025 nM T34296 CP9WG5 10389610 IC50 = 1.8 nM T34296 CY2G0R 10391428 Ki > 5025 nM T34296 C8O1XU 10392082 IC50 = 0.1 nM T34296 C8Y7EZ 10393391 IC50 = 28 nM T34296 CFKA79 10395015 Ki = 653 nM T34296 C1SJ4K 10435554 IC50 = 20 nM T34296 C7XE1L 10437629 IC50 = 4000 nM T34296 C5WV1N 10439082 Ki = 442 nM T34296 C54UDR 10453826 IC50 = 400 nM T34296 C8M9FE 10462640 Ki = 15700 nM T34296 CX38EB 10467565 IC50 = 460 nM T34296 CNQZ36 10483139 Ki = 0.66 nM T34296 C9XC8Y 10493383 IC50 = 79 nM T34296 C6KD0A 10498747 IC50 = 1 nM T34296 CZ2UY0 10502046 IC50 = 2.3 nM T34296 C36OMW 10502172 IC50 = 1 nM T34296 C5V8HJ 10502382 IC50 = 0.8 nM T34296 CJZ5T8 10502487 IC50 > 10000 nM T34296 CSN17G 10502708 IC50 = 0.9 nM T34296 CBNM82 10503128 IC50 < 0.4 nM T34296 C9LJR5 10503737 IC50 = 137 nM T34296 C5Y4IA 10504081 IC50 = 478 nM T34296 C2C7TE 10504472 IC50 < 0.5 nM T34296 CH6S8Y 10505729 IC50 > 10000 nM T34296 C6D7JF 10506147 IC50 = 36 nM T34296 C7S0DB 10506158 IC50 = 24 nM T34296 CBT12Q 10522080 IC50 = 0.7 nM T34296 CC2F5Y 10522311 IC50 = 1 nM T34296 CZ36JW 10523383 IC50 = 580 nM T34296 CQEH42 10524134 IC50 < 0.5 nM T34296 CYU87N 10524260 IC50 < 0.4 nM T34296 COT07L 10525329 IC50 = 8 nM T34296 C61GSD 10525562 IC50 = 2.5 nM T34296 C14XUW 10526101 IC50 = 3 nM T34296 CJK6G1 10526509 IC50 < 0.1 nM T34296 CWLD37 10526788 IC50 = 1 nM T34296 CHS9Q5 10527785 IC50 = 0.8 nM T34296 CJ0D7G 10528505 IC50 = 1.3 nM T34296 CYGU41 10529315 IC50 = 2137.96 nM T34296 CO2R0P 10544323 IC50 = 21 nM T34296 C4PK0U 10549114 IC50 = 1 nM T34296 C4TA1K 10549256 IC50 < 0.4 nM T34296 CHCI01 10549577 IC50 = 0.4 nM T34296 C2HJ1U 10549764 IC50 = 1 nM T34296 CRHP20 10550304 IC50 = 1.5 nM T34296 C7WQ5Z 10550399 IC50 = 2 nM T34296 CNQ75F 10551139 IC50 = 21 nM T34296 CCH0K3 10551483 IC50 = 2.1 nM T34296 CC2FM6 10551489 IC50 > 1600 nM T34296 C5UD0A 10551910 IC50 = 21 nM T34296 CI8XG0 10554869 IC50 = 7 nM T34296 CT7O9M 10569678 IC50 = 11 nM T34296 C8RWE4 10569743 IC50 = 105 nM T34296 CE14GM 10570702 IC50 = 6 nM T34296 CS9Y3Q 10573446 IC50 = 0.5 nM T34296 C61IUN 10574937 IC50 = 3.3 nM T34296 C1KH7E 10578728 IC50 = 154 nM T34296 CIUO27 10593253 IC50 = 1 nM T34296 CUTS47 10594564 IC50 = 37 nM T34296 CN4Y6H 10594565 IC50 = 53 nM T34296 CYNC76 10596158 IC50 = 10 nM T34296 C0R8ND 10599533 IC50 < 0.4 nM T34296 CQCW86 10599579 IC50 < 0.4 nM T34296 CW18QK 10599594 IC50 = 0.4 nM T34296 CR1JI4 10600645 IC50 = 0.9 nM T34296 C6RH4O 10601640 IC50 = 4.5 nM T34296 CG32FM 10613145 IC50 = 18 nM T34296 CZD9B3 10617580 IC50 = 1.9 nM T34296 CL02BO 10618584 IC50 = 16 nM T34296 C0JGS3 10621776 IC50 = 3 nM T34296 CL5QN9 10622296 IC50 = 1.9 nM T34296 CL62YC 10622822 IC50 = 9.2 nM T34296 CZJB31 10622970 IC50 = 2.9 nM T34296 CL67UQ 10623250 IC50 = 478.63 nM T34296 CGB29T 10625771 IC50 = 0.5 nM T34296 C98KGO 10625860 IC50 = 3.2 nM T34296 C8UY9P 10639050 IC50 > 30000 nM T34296 C7KGM3 10642071 IC50 = 0.7 nM T34296 CWRY91 10642128 IC50 = 3.6 nM T34296 CI2QB9 10642965 IC50 < 1 nM T34296 C2O1XM 10647817 IC50 = 2.8 nM T34296 C5RWF4 10648802 IC50 = 2 nM T34296 C6S1KA 10649216 IC50 > 10000 nM T34296 C27QHB 10663143 IC50 = 1.7 nM T34296 C97KZU 10665624 IC50 = 43 nM T34296 CF0E6H 10668745 IC50 = 23 nM T34296 CAI72H 10670246 IC50 = 0.7 nM T34296 CY6QC1 10670819 IC50 = 4.1 nM T34296 CPG5O2 10671155 IC50 = 2.4 nM T34296 C17LYV 10672346 IC50 = 48.98 nM T34296 CMU74I 10672857 IC50 = 269.15 nM T34296 CXTP56 10688727 IC50 < 0.5 nM T34296 C0OJ9C 10689683 IC50 = 5 nM T34296 CSA80H 10692194 IC50 = 1 nM T34296 CS5CL7 10692307 IC50 = 0.5 nM T34296 CR5KF8 10692994 IC50 = 710 nM T34296 CDI12G 10693559 IC50 = 1.3 nM T34296 CB70DA 10693592 IC50 = 0.9 nM T34296 CVML68 10693881 IC50 = 1 nM T34296 CZGC63 10695865 IC50 = 102.33 nM T34296 CW6CF7 10696226 IC50 = 1 nM T34296 C6MWX8 10696713 IC50 = 26.92 nM T34296 C1YFC3 10696977 IC50 = 223.87 nM T34296 C4BME8 10697140 IC50 = 254 nM T34296 CG38ZD 10714323 IC50 = 27 nM T34296 C4IWF2 10714988 IC50 = 1 nM T34296 CO9KV7 10715115 IC50 = 0.3 nM T34296 CE1D6G 10716217 IC50 = 0.2 nM T34296 C0ZX6T 10717308 IC50 = 5 nM T34296 C7OSW8 10718200 IC50 < 0.4 nM T34296 C35MRE 10719092 IC50 = 0.4 nM T34296 CVW81M 10719595 IC50 = 114.82 nM T34296 C4J1WN 10721454 IC50 = 2 nM T34296 CI4SQ2 10732349 IC50 = 500 nM T34296 C51DZG 10737732 IC50 = 48 nM T34296 C1LS5U 10738104 IC50 = 1 nM T34296 CL74TG 10738165 IC50 < 0.4 nM T34296 C76ANK 10739335 IC50 = 1 nM T34296 C0T2VK 10740460 IC50 = 1.698 nM T34296 CKJD45 10741133 IC50 = 650 nM T34296 CL64BU 10741592 IC50 < 0.4 nM T34296 C4MQ8L 10742072 IC50 < 0.4 nM T34296 CKX5R3 10742142 IC50 = 21.88 nM T34296 CHW23E 10742387 IC50 = 2.7 nM T34296 CCH94Q 10743507 IC50 = 1.3 nM T34296 C9ILP3 10745718 IC50 = 13 nM T34296 CE09PI 10757715 IC50 = 5 nM T34296 C0BAE9 10763583 IC50 = 2037 nM T34296 C68THN 10763851 IC50 < 0.2 nM T34296 CAG53Y 10764489 IC50 = 5.6 nM T34296 C0ZJB9 10764600 IC50 = 57 nM T34296 CJE76M 10764871 IC50 = 0.7 nM T34296 CQ0KM4 10765140 IC50 < 0.4 nM T34296 C3P2TS 10766036 IC50 = 144.54 nM T34296 CN6P1J 10766950 IC50 = 17 nM T34296 CWR5Z3 10767105 IC50 = 58.88 nM T34296 CR4I1E 10767157 IC50 = 125.89 nM T34296 C7Q2EM 10767236 IC50 = 2 nM T34296 CQ7J4I 10769007 IC50 = 344 nM T34296 C2FA7J 10787997 IC50 = 1 nM T34296 C16XQR 10788211 IC50 = 0.4 nM T34296 C0DFB9 10788617 IC50 < 0.2 nM T34296 CNAE08 10788733 IC50 = 7 nM T34296 CXQD12 10789326 IC50 = 1659.59 nM T34296 CKV2O8 10789493 IC50 = 0.7 nM T34296 C45UGJ 10789671 IC50 < 0.4 nM T34296 C9NZ4W 10789711 IC50 = 1 nM T34296 CHWG02 10790787 IC50 = 88 nM T34296 CWCD73 10805054 IC50 = 4 nM T34296 C1WZ4S 10805349 IC50 = 1 nM T34296 CN8I3Z 10808172 IC50 = 11 nM T34296 CT1AI4 10810573 IC50 = 2 nM T34296 CV3ZA5 10812444 IC50 = 54 nM T34296 CZB7L2 10812929 IC50 < 1 nM T34296 C4TF0K 10813874 IC50 = 0.1 nM T34296 CCIL63 10813879 IC50 < 0.4 nM T34296 CIUN51 10814028 IC50 = 144.54 nM T34296 CS7BY4 10816934 IC50 = 4 nM T34296 CX2E1C 10829071 IC50 = 0.5 nM T34296 C3AI5Z 10831752 IC50 = 150 nM T34296 CLK9P7 10832592 IC50 = 18.4 nM T34296 CF50HD 10832925 IC50 = 26 nM T34296 C5OG4U 10833497 IC50 = 102 nM T34296 CH90ZB 10834348 IC50 = 4.3 nM T34296 C48PYQ 10836923 IC50 = 1.4 nM T34296 CH8OV4 10837276 IC50 = 2.5 nM T34296 CF40VH 10837557 IC50 = 0.8 nM T34296 CY4J9A 10838149 IC50 = 0.9 nM T34296 CA76MU 10840059 IC50 = 2754.23 nM T34296 CN5MJ6 10853865 IC50 = 3390 nM T34296 C3UCL2 10854279 IC50 = 9 nM T34296 CBQ70P 10874312 IC50 = 16.2 nM T34296 CXY47P 10875332 IC50 = 2.8 nM T34296 C3AY8O 10885569 IC50 = 31 nM T34296 CAU0I3 10885834 IC50 = 2.399 nM T34296 CG1I4Y 10886343 IC50 = 2 nM T34296 CF5L1R 10886549 IC50 = 4 nM T34296 CPJ0I8 10896934 IC50 = 808 nM T34296 CU7YE0 10896986 IC50 = 0.5 nM T34296 CX93MR 10907320 IC50 = 27 nM T34296 CAH70N 10914350 IC50 = 37 nM T34296 CF9NT3 10914471 IC50 = 141 nM T34296 CGI2T1 10928606 IC50 = 275 nM T34296 CXHA75 10928874 IC50 = 5.37 nM T34296 C40PRC 10929100 IC50 = 19 nM T34296 CXY4L6 10929354 IC50 = 417 nM T34296 CDSQ41 10929404 IC50 = 391 nM T34296 C4JC9O 10930047 IC50 = 3.02 nM T34296 CLIR35 10938505 IC50 = 2 nM T34296 CWO29J 10940364 IC50 = 80 nM T34296 C9YOU4 10951375 IC50 = 14 nM T34296 CJI1G0 10951750 IC50 = 0.8 nM T34296 C3K1BL 10959017 IC50 = 11 nM T34296 C5ZV9Q 10962137 IC50 = 11 nM T34296 CR9J5B 10983887 IC50 = 5.1 nM T34296 CSI5G1 10992109 IC50 = 6 nM T34296 CCX0L6 10994350 IC50 = 5.1 nM T34296 C9C8SA 11001101 IC50 = 64 nM T34296 C4PNK3 11006191 IC50 = 407 nM T34296 CS4FL3 11012667 IC50 = 12 nM T34296 C5JE9G 11014504 IC50 = 14 nM T34296 C9WPH7 11016072 Ki > 15000 nM T34296 CBE68H 11016073 Ki > 15000 nM T34296 CG2DK0 11016448 IC50 = 1 nM T34296 CF30UR 11016519 IC50 = 5.3 nM T34296 CODQ51 11016616 IC50 = 0.3981 nM T34296 C6IHF5 11026991 IC50 > 100 nM T34296 C23KPN 11050468 IC50 = 4.5 nM T34296 C9RU4I 11059620 IC50 = 29.5 nM T34296 C1N5PT 11070986 IC50 = 13.8 nM T34296 C18EIZ 11071831 IC50 = 1 nM T34296 CM9EP0 11077031 IC50 = 188 nM T34296 C5MUD2 11078779 IC50 = 85 nM T34296 CG0A4C 11081333 IC50 = 32 nM T34296 C05MUK 11081992 IC50 = 3.2 nM T34296 CS29GX 11091928 IC50 = 15 nM T34296 C16WBE 11092175 IC50 = 12 nM T34296 CE8V9B 11092295 IC50 = 11.8 nM T34296 CR8ZA7 11092551 IC50 = 195 nM T34296 CX69YN 11093502 IC50 = 1.6 nM T34296 C6CLV8 11101735 IC50 = 319 nM T34296 CR4V2D 11101785 Ki = 620 nM T34296 C8CK3E 11102531 IC50 = 66 nM T34296 CEAI92 11112993 IC50 = 1 nM T34296 CY1SR9 11113744 IC50 = 140 nM T34296 CB2I5K 11123701 IC50 = 55 nM T34296 C8YVE5 11123989 IC50 = 13 nM T34296 CNBG53 11124956 IC50 = 2.3 nM T34296 C2YBQ7 11134935 IC50 = 6.9 nM T34296 C8DMW5 11135133 IC50 = 1.8 nM T34296 CD3N8B 11135304 IC50 = 23 nM T34296 CPO02F 11142863 IC50 = 1.4 nM T34296 C3V4ZX 11143285 IC50 = 12 nM T34296 C9H1CW 11156691 IC50 = 2.3 nM T34296 CMKT17 11168614 IC50 = 8 nM T34296 C63CLD 11169065 IC50 = 220 nM T34296 CVI3F8 11188429 IC50 = 3687 nM T34296 CPA84O 11192618 IC50 = 32 nM T34296 CO5VN2 11201367 IC50 > 10000 nM T34296 CET3R7 11201814 IC50 = 284 nM T34296 C43ONW 11202395 Ki = 4314 nM T34296 CO87YZ 11215538 IC50 = 19 nM T34296 CIZW31 11226189 IC50 = 4.3 nM T34296 C72UCB 11233687 IC50 = 68 nM T34296 CS15WB 11236105 IC50 = 38 nM T34296 CJZ3P6 11257884 Ki = 0.54 nM T34296 CD1FT8 11258906 IC50 = 7 nM T34296 CJM90S 11259332 IC50 = 6.72 nM T34296 C2OJ8Q 11272747 IC50 = 9.5 nM T34296 CC62RY 11279665 IC50 = 38 nM T34296 CJX60I 11284255 IC50 = 6.5 nM T34296 C6LJM4 11284404 IC50 = 3 nM T34296 CP17ID 11284983 IC50 = 2.3 nM T34296 C1IW7N 11292680 IC50 = 4.1 nM T34296 C8C5AV 11294179 Ki > 10000 nM T34296 CLH50U 11318841 IC50 = 7.1 nM T34296 C1SN8I 11319030 IC50 = 3.2 nM T34296 C91LBZ 11319396 IC50 = 58 nM T34296 C48JVH 11327633 IC50 = 2200 nM T34296 C9FW7I 11330706 IC50 = 15 nM T34296 C0XR3B 11330861 IC50 = 11 nM T34296 C49CDU 11335940 IC50 = 970 nM T34296 CQH57S 11342435 IC50 = 1.8 nM T34296 CZ8B0D 11349945 Ki < 5 nM T34296 CYAK73 11353754 IC50 = 3 nM T34296 CTQK48 11373358 Ki > 5025 nM T34296 C5KU3Z 11376005 IC50 = 6.1 nM T34296 CL8QO7 11382562 IC50 = 900 nM T34296 CNZ0T5 11386918 IC50 = 5 nM T34296 CEM0A7 11387990 IC50 = 25 nM T34296 C9KVB7 11394505 IC50 = 32 nM T34296 C9ABX8 11397130 Ki > 5025 nM T34296 CF78WB 11398934 IC50 = 7.8 nM T34296 C2EUO5 11417011 IC50 > 10000 nM T34296 C30PFC 11421763 IC50 = 6.4 nM T34296 CK95HW 11429232 Ki = 1.2 nM T34296 C01FLQ 11441438 Ki < 5 nM T34296 C5NAJ3 11449819 IC50 = 72 nM T34296 COS67B 11456566 IC50 = 2.1 nM T34296 C96DRO 11466734 IC50 = 3.7 nM T34296 C7QF0G 11467517 IC50 = 13 nM T34296 C1KP2Q 11473879 Ki > 5025 nM T34296 C5QEZ8 11483818 IC50 = 18 nM T34296 CX9IY2 11496709 IC50 = 95.6 nM T34296 C3RJ8Z 11496896 IC50 = 4 nM T34296 C6HU4N 11503290 IC50 = 28 nM T34296 CJ46KN 11508259 Ki = 3.6 nM T34296 CWS35C 11510523 IC50 = 13600 nM T34296 C5VUM2 11517085 Ki = 510 nM T34296 CQ9E6J 11519157 IC50 = 2.6 nM T34296 C5MO0U 11526826 IC50 = 15 nM T34296 C9Y6LH 11533683 IC50 = 4440 nM T34296 C5V8UA 11540282 IC50 = 184 nM T34296 C1NZB9 11548265 IC50 = 1.1 nM T34296 CC4GZ0 11554178 IC50 = 2.69 nM T34296 CE3HA6 11556698 Ki = 4000 nM T34296 CNZV95 11561070 IC50 = 16.4 nM T34296 CCW1B8 11569185 IC50 = 5.4 nM T34296 CW5A4S 11569716 IC50 = 2.2 nM T34296 CL9K7T 11583525 IC50 = 8.5 nM T34296 CTQ87G 11599024 IC50 = 4560 nM T34296 CVGC49 11603611 Ki = 2 nM T34296 C7L1NB 11604052 IC50 = 184 nM T34296 C8IWM1 11605689 IC50 = 1.2 nM T34296 C0VCJ8 11613810 IC50 = 6.3 nM T34296 CC2YD9 11618883 IC50 = 4.24 nM T34296 C9EOY7 11619541 IC50 = 11 nM T34296 CCBS59 11634234 IC50 = 157 nM T34296 CNY92D 11640694 Ki = 7000 nM T34296 C1U3EX 11656290 IC50 = 9.8 nM T34296 C3LZP9 11662242 IC50 = 120 nM T34296 CPIN09 11668791 IC50 = 19.3 nM T34296 CRF7V9 11691964 IC50 = 1.1 nM T34296 C3U6ZR 11697504 Ki = 20000 nM T34296 C1NGT6 11698000 IC50 = 18 nM T34296 C4BGI2 11698938 IC50 = 1336 nM T34296 C2BJ3X 11716217 Ki = 12860 nM T34296 CCD93H 11730086 Ki = 180 nM T34296 C7CED0 11733417 IC50 = 791 nM T34296 CI0KL2 11733573 IC50 = 11 nM T34296 C27SBC 11734162 IC50 = 1 nM T34296 C6HV8Z 11752434 IC50 = 3 nM T34296 CG8U3H 11753351 IC50 = 25 nM T34296 CO8QT0 11753905 Ki = 490 nM T34296 CJ4G5D 11754907 IC50 = 18.1 nM T34296 CE6OS0 11755521 IC50 = 1.288 nM T34296 CL4NF5 11756420 IC50 = 0.11 nM T34296 CUC9R5 11758082 IC50 = 0.7 nM T34296 C2KU3D 11760296 IC50 = 6 nM T34296 CKM6P2 11795228 IC50 = 4.2 nM T34296 CCSD72 11795621 IC50 = 2.1 nM T34296 C46KHU 11796490 IC50 = 1.3 nM T34296 C47OIA 11797154 IC50 = 0.8 nM T34296 CCD4W2 11797992 IC50 = 1.1 nM T34296 CHQR96 11798386 IC50 = 0.2 nM T34296 C2YD4N 11809525 IC50 = 39 nM T34296 C1NRV6 11811437 IC50 = 9 nM T34296 CQ9HE2 11811551 IC50 = 264 nM T34296 CLW3F1 11812791 IC50 = 55.3 nM T34296 CH3SV6 11813493 IC50 = 296 nM T34296 C7BK5P 11825105 IC50 = 0.4 nM T34296 CKEM29 11827006 IC50 = 162 nM T34296 C4XR5G 11963536 IC50 = 2277 nM T34296 C02BWA 11967143 Ki > 2000 nM T34296 CB80OT 12000718 IC50 = 0.03 nM T34296 C43PJZ 12000720 IC50 = 1.3 nM T34296 CUQM03 12074753 IC50 = 1100 nM T34296 CKND02 12074756 IC50 = 1100 nM T34296 C4I1TJ 12074757 IC50 = 3700 nM T34296 CJ8W2C 12074758 IC50 = 800 nM T34296 C0K8ZX 12404978 IC50 > 500000 nM T34296 CB1F2E 12971983 IC50 = 825 nM T34296 CJY6X7 12971984 IC50 = 281 nM T34296 CZYE40 12971985 IC50 = 331 nM T34296 C8TH1O 14177156 IC50 > 500000 nM T34296 CKN3R1 15430588 IC50 = 291 nM T34296 C63MFQ 15435266 IC50 = 7 nM T34296 CZ0NL1 15484680 IC50 = 16 nM T34296 C70TDZ 15503645 IC50 = 136 nM T34296 C16TEM 15516782 IC50 = 18 nM T34296 CV1HA9 15516783 IC50 = 2 nM T34296 CEKN36 15520981 IC50 = 0.35 nM T34296 CXUG10 15546245 IC50 = 50 nM T34296 CU7CM3 15551877 IC50 = 56 nM T34296 C2WHJ4 15859211 IC50 = 555 nM T34296 C5FA3L 15871222 IC50 = 12 nM T34296 C6R1LD 15985818 IC50 = 96 nM T34296 C6HM9P 16069178 IC50 = 0.034 nM T34296 CS46XU 16126723 IC50 = 1.6 nM T34296 CC1K9A 16651091 IC50 > 398107.17 nM T34296 CT40DY 16651117 IC50 = 31622.78 nM T34296 C91EXN 16655061 IC50 = 259 nM T34296 CY7DO3 16718635 IC50 = 0.062 nM T34296 CBIH04 16719299 IC50 = 0.024 nM T34296 CP82IZ 16719300 IC50 = 0.054 nM T34296 CQS0F5 16719301 IC50 = 0.036 nM T34296 C97REC 16719303 IC50 = 0.14 nM T34296 C75XDI 16730519 IC50 > 5000 nM T34296 C2W1VA 16739287 Ki = 1200 nM T34296 C3S2TQ 17754305 IC50 = 2920 nM T34296 C6O3KA 17781194 IC50 = 0.53 nM T34296 CIR7S8 17866387 IC50 = 3 nM T34296 CL1H9W 17866459 IC50 = 20 nM T34296 C9RNH3 17866675 IC50 = 12 nM T34296 CCGR13 17897285 IC50 = 3 nM T34296 C2ZAX1 18002715 Ki > 5000 nM T34296 C12UGK 18002722 Ki = 503 nM T34296 C0IYW8 18002726 Ki > 5000 nM T34296 C8N1DM 18002729 Ki = 754 nM T34296 CCG96A 18002736 Ki = 955 nM T34296 C5MLG1 18002745 Ki > 5000 nM T34296 CXT4H2 18002752 Ki > 5000 nM T34296 C26WHK 18002758 Ki = 1708 nM T34296 CV90XS 18002764 Ki > 5000 nM T34296 C8KPM7 18002765 Ki > 5000 nM T34296 CMJ0K3 18002771 Ki > 5000 nM T34296 C2CO9Z 18002775 Ki > 5000 nM T34296 CK8FS7 18173159 IC50 = 101 nM T34296 CX10BM 18173179 IC50 = 65 nM T34296 CQO70Y 18173222 IC50 = 485 nM T34296 C6AW0H 18365436 IC50 = 17 nM T34296 C1QIU4 18368941 IC50 = 15000 nM T34296 C0VJG4 18368975 IC50 = 15000 nM T34296 CI53DY 18379040 Ki > 5025 nM T34296 CB1U5T 18379077 Ki > 5025 nM T34296 CSX97G 18379115 Ki > 5025 nM T34296 CJHL25 18379123 Ki > 5025 nM T34296 CR0B8G 18379149 Ki > 5025 nM T34296 CS4V5K 18379187 Ki > 5025 nM T34296 CCTY94 18379210 Ki > 5025 nM T34296 CA6K5S 18379235 Ki > 5025 nM T34296 CCSK49 18379254 Ki > 5025 nM T34296 CP4T7S 18379435 Ki > 5025 nM T34296 C9Y5GX 18379443 Ki > 5025 nM T34296 CS2H6J 18396836 IC50 = 250 nM T34296 C1WUJ0 18512732 IC50 < 1000 nM T34296 CA0JF9 18512733 IC50 = 15000 nM T34296 C8EIC6 18512737 IC50 = 5900 nM T34296 C50AEZ 18616892 IC50 = 1.7 nM T34296 CRI35F 19366819 IC50 = 1500 nM T34296 CC4KN8 19366830 IC50 = 1 nM T34296 CS70KY 19366867 IC50 = 0.4 nM T34296 CE73XW 19366873 IC50 = 700 nM T34296 CK8MP3 20620240 Ki = 0.13 nM T34296 CPC4G6 20620273 Ki = 2 nM T34296 C26UJT 20620561 IC50 = 0.9 nM T34296 C2E3CY 20620614 IC50 = 0.2 nM T34296 CVEX54 20620688 IC50 = 0.9 nM T34296 CV1SD8 20620714 IC50 = 0.2 nM T34296 C3GAC4 20620715 IC50 = 3.3 nM T34296 C7QV8K 20620757 IC50 = 1.6 nM T34296 CVO73Y 20620827 IC50 = 8.2 nM T34296 CQ14NY 20620831 IC50 = 8 nM T34296 C5RQ8A 20620860 IC50 = 1.7 nM T34296 CPK09X 20651316 IC50 = 1 nM T34296 C30EAU 20651317 IC50 = 305 nM T34296 C48TWB 20728102 IC50 > 5000 nM T34296 C18RXS 20735191 IC50 < 0.1 nM T34296 C4I1OM 20735209 IC50 = 9 nM T34296 CF1CK9 20735364 IC50 = 1 nM T34296 C09JTR 21130554 IC50 = 0.4 nM T34296 CW1JS2 21130555 IC50 = 24000 nM T34296 C6VP1T 21130556 IC50 = 0.3 nM T34296 C15UGO 21130558 IC50 = 24 nM T34296 C9H3IG 21130559 IC50 = 1.6 nM T34296 C8Q2OD 21130561 IC50 = 2.4 nM T34296 C25FAD 21130562 IC50 = 0.6 nM T34296 C3FAU5 21130572 IC50 = 600 nM T34296 C19AEV 21130574 IC50 = 400 nM T34296 CW2Q5A 21130590 IC50 = 160 nM T34296 C9HMC0 21130591 IC50 = 161 nM T34296 CM92DX 21304705 IC50 = 9 nM T34296 CJ0Y9V 21304706 IC50 = 7 nM T34296 C5X1YM 21304708 IC50 = 11 nM T34296 C0Z3LD 21304710 IC50 = 1 nM T34296 C8F5AH 21310747 IC50 = 26 nM T34296 CG18HB 21310751 IC50 = 19 nM T34296 CEW0M3 21310753 IC50 = 11 nM T34296 CC2L1Z 21310756 IC50 = 959 nM T34296 C0T2QX 21310757 IC50 = 24 nM T34296 CWM7F2 21310775 IC50 = 138 nM T34296 CNEW70 21310777 IC50 = 50 nM T34296 CY12PI 21310778 IC50 = 42 nM T34296 CV10FJ 21310779 IC50 = 134.9 nM T34296 CPT4E5 21310780 IC50 = 982 nM T34296 CJ2U7K 21310781 IC50 = 728 nM T34296 C5SG2L 21310789 IC50 = 84 nM T34296 C3TI6Y 21310790 IC50 = 1 nM T34296 C87BMF 21310824 IC50 = 14 nM T34296 C26IPQ 21310829 IC50 = 11 nM T34296 CIB1X5 21310851 IC50 = 43 nM T34296 C6OZL3 21310926 IC50 = 113 nM T34296 C72BVA 21310934 IC50 = 717 nM T34296 CUJ6A1 21310984 IC50 = 137 nM T34296 C96REO 21584504 IC50 = 15 nM T34296 C8N6DH 21931010 IC50 = 0.53 nM T34296 CA6E9I 21931045 IC50 = 7.5 nM T34296 CN16ZT 21931049 IC50 = 0.63 nM T34296 C8IBZ2 21931061 IC50 = 0.4 nM T34296 CVS02H 21931065 IC50 = 1.6 nM T34296 CM9XW7 21931067 IC50 = 0.35 nM T34296 C27BZI 21931069 IC50 = 7.8 nM T34296 CO46GR 21931088 IC50 = 3.4 nM T34296 CS2KZ5 21931099 IC50 = 2.4 nM T34296 C7PQU4 21931103 IC50 = 6.1 nM T34296 CLQ58R 21931105 IC50 = 0.34 nM T34296 CWCN52 21931106 IC50 = 1 nM T34296 CX6QD0 21931115 IC50 = 12 nM T34296 COJ2R8 21931118 IC50 = 0.84 nM T34296 C94BWM 21931138 IC50 = 0.46 nM T34296 CIC4S9 22004232 IC50 = 7 nM T34296 C5FWN2 22248619 IC50 = 77 nM T34296 CH6U1G 22338710 IC50 = 75 nM T34296 CO91AD 22341241 Ki > 5025 nM T34296 CJW3E0 22482219 IC50 = 194 nM T34296 CE5DH1 22484408 IC50 = 1.8 nM T34296 CZT05X 22484417 Ki = 1.6 nM T34296 CZT64B 22484431 Ki = 1.5 nM T34296 C1O7RC 22485248 IC50 = 70 nM T34296 CAM10T 22485252 IC50 = 0.8 nM T34296 CBJS34 22485260 IC50 < 0.1 nM T34296 C9MU7N 22485263 IC50 = 6 nM T34296 CEGJ03 22485276 IC50 = 2.9 nM T34296 C7VB8G 22485289 IC50 = 0.3 nM T34296 CNB02I 22485291 IC50 = 0.1 nM T34296 CAY3N6 22485292 IC50 = 2.7 nM T34296 C94OCJ 22485302 IC50 = 0.25 nM T34296 C3YL5X 22485311 IC50 = 0.25 nM T34296 C80RSQ 22485314 IC50 = 0.2 nM T34296 CWA03L 22485327 IC50 = 0.3 nM T34296 C6JRW5 22485340 IC50 = 0.1 nM T34296 C5JZF1 22485344 IC50 = 0.8 nM T34296 CI7MY5 22485346 IC50 = 0.25 nM T34296 CI1YL7 22485347 IC50 = 0.2 nM T34296 C25OBD 22485356 IC50 = 0.45 nM T34296 C7I0EW 22485367 IC50 = 0.3 nM T34296 CL64TJ 22485368 IC50 = 0.6 nM T34296 CT4GF9 22485381 IC50 = 27.7 nM T34296 C27NDB 22485386 IC50 = 1.2 nM T34296 CTJ9I3 22485392 IC50 = 0.5 nM T34296 C3MG9P 22485396 IC50 = 1.9 nM T34296 CZY10U 22485408 IC50 = 5.5 nM T34296 C89AGT 22485413 IC50 = 0.6 nM T34296 C03NLM 22485417 IC50 = 0.1 nM T34296 C8GHU9 22485432 IC50 = 0.5 nM T34296 CIN18B 22598309 IC50 = 15.1 nM T34296 C2X3VB 22598316 IC50 = 1.57 nM T34296 C9BT5F 22626996 IC50 = 114 nM T34296 C7ITG0 22644780 IC50 = 20.89 nM T34296 CIQ76F 22644837 IC50 = 5 nM T34296 CYJ48I 22644895 IC50 = 36 nM T34296 CQB36V 22644965 IC50 = 4 nM T34296 CVM1O6 22644970 IC50 = 7 nM T34296 C0K1GE 22645081 IC50 = 20 nM T34296 C2Q4XK 22707806 IC50 = 0.2 nM T34296 CD4Z6P 22707833 IC50 = 20 nM T34296 CMYK90 22707860 IC50 < 0.1 nM T34296 CDQ12R 22712799 IC50 = 100000 nM T34296 CX40LP 22712801 IC50 = 75000 nM T34296 CVF9M4 22922043 IC50 = 42520 nM T34296 CIYA45 22985930 IC50 = 0.1 nM T34296 CF75MS 23017979 IC50 = 25000 nM T34296 CQJ3S4 23018008 IC50 = 7000 nM T34296 C9IW3E 23433373 IC50 = 6700 nM T34296 C4VG8C 23506747 IC50 = 433 nM T34296 CK97AT 23506779 IC50 = 68 nM T34296 CP94QR 23506783 IC50 = 11 nM T34296 CX32YK 23513795 IC50 = 10 nM T34296 C6IZ1S 23513821 IC50 = 69 nM T34296 CPNM93 23513825 IC50 = 59 nM T34296 CML90Q 23513831 IC50 = 54 nM T34296 C87RTM 23513845 IC50 = 327 nM T34296 CNSU58 23513850 IC50 = 135 nM T34296 C4R2AJ 23625454 IC50 = 3199 nM T34296 CD3U8A 23627203 Ki = 1700 nM T34296 CL24JR 23655078 IC50 = 470 nM T34296 COIZ43 23655713 IC50 = 9140 nM T34296 CURM98 23655714 IC50 > 100000 nM T34296 CO90JC 23655717 IC50 > 100000 nM T34296 C56NMQ 23655910 IC50 = 34000 nM T34296 C9QZX5 23655911 IC50 = 3260 nM T34296 CA8W3K 23656106 IC50 = 384 nM T34296 CU4R7T 23656291 IC50 = 11 nM T34296 CVZ2M1 23656293 IC50 = 10 nM T34296 CL5C1I 23656295 IC50 = 59 nM T34296 CZP12E 23656450 IC50 = 24 nM T34296 CA2PY5 23657418 IC50 = 10 nM T34296 CN9TY1 23657419 IC50 = 1340 nM T34296 C9FHZ1 23657421 IC50 = 50 nM T34296 CY9LF1 23657422 IC50 = 0.9 nM T34296 C28SPW 23657691 IC50 = 14000 nM T34296 CVJ1T7 23657695 IC50 = 41000 nM T34296 CAL05Q 23657697 IC50 = 30000 nM T34296 C3TWS6 24178109 Ki = 2.7 nM T34296 C35QME 24742028 IC50 = 0.8 nM T34296 CXEP14 24754176 IC50 > 100000 nM T34296 CSQ9E4 24754248 IC50 > 22000 nM T34296 CX16GL 24754251 IC50 > 100000 nM T34296 COY8K0 24754252 IC50 > 100000 nM T34296 CG3J2L 24768528 IC50 = 860 nM T34296 CQCJ17 24768595 IC50 = 0.2 nM T34296 CUS47E 24795059 IC50 = 65 nM T34296 CDRP74 24801536 IC50 = 1.61 nM T34296 CI61SG 24801701 IC50 = 31.1 nM T34296 C18FRG 24807817 IC50 = 55000 nM T34296 CW3X0F 24852010 IC50 = 6.8 nM T34296 C6YPS8 24852048 IC50 = 2.5 nM T34296 C4LXM8 24860420 IC50 = 1600 nM T34296 CK0CI6 24860421 IC50 = 1038 nM T34296 CZI59C 24860423 IC50 = 2075 nM T34296 CE29HI 24860424 IC50 = 6882 nM T34296 CT10JE 24860425 IC50 = 772 nM T34296 CRC98J 24860426 IC50 = 584 nM T34296 C8MKR0 24860427 IC50 = 2476 nM T34296 C3S6DX 24860428 IC50 = 30 nM T34296 C2LNE4 24860429 IC50 = 2912 nM T34296 CF4D0X 24860430 IC50 = 12000 nM T34296 C4FI5C 24901479 IC50 = 62 nM T34296 C6F0ZP 24901485 IC50 = 2.6 nM T34296 C4SP3O 24936157 IC50 = 0.19 nM T34296 CBUA83 24936183 IC50 = 7.3 nM T34296 C0EA5F 24936382 IC50 = 0.062 nM T34296 CB94KU 24958549 IC50 > 100000 nM T34296 CU3W7Y 24960377 IC50 > 200000 nM T34296 CNCA57 25004194 Ki = 4.677 nM T34296 CAQ9Z1 25022681 Ki > 5025 nM T34296 CA86UE 25049752 Ki = 2.2 nM T34296 C82NLV 25049754 Ki = 46 nM T34296 C6QFV4 25049756 Ki = 42 nM T34296 C4HVF2 25064051 IC50 = 93 nM T34296 C64BZH 25064052 IC50 = 1.22 nM T34296 CZ2TG0 25064053 IC50 = 1135 nM T34296 C3S8OA 25064054 IC50 = 277 nM T34296 CA64KF 25064283 IC50 = 456 nM T34296 C94MXR 25064485 IC50 = 200 nM T34296 CD9T2O 25064489 IC50 = 809 nM T34296 C3BC9Z 25064704 IC50 = 1286 nM T34296 C23TDS 25064904 IC50 = 632 nM T34296 C54MLN 25064905 IC50 = 56 nM T34296 C7T2UO 25064906 IC50 = 334 nM T34296 C16AIC 25064907 IC50 = 1353 nM T34296 CL9N8I 25064908 IC50 = 147 nM T34296 CJP30U 25065108 IC50 = 235 nM T34296 CMZV31 25065109 IC50 = 217 nM T34296 C03NHX 25065111 IC50 = 23 nM T34296 CE72DR 25065318 IC50 = 500 nM T34296 CEK1Y2 25065514 IC50 = 109 nM T34296 C3F5LH 25065515 IC50 = 500 nM T34296 CB0Z5P 25065946 IC50 = 1100 nM T34296 CJWD41 25066149 IC50 = 25000 nM T34296 CI4A7E 25066153 IC50 = 6000 nM T34296 CN9UM1 25066154 IC50 > 25000 nM T34296 CEU95V 25066364 IC50 > 25000 nM T34296 C0FJK5 25066365 IC50 > 25000 nM T34296 CZY4L8 25066366 IC50 > 25000 nM T34296 C2ZS5J 25066563 IC50 = 65 nM T34296 C6CMU0 25066564 IC50 = 180 nM T34296 CZO08G 25066566 IC50 = 100 nM T34296 C58KNZ 25066763 IC50 = 10 nM T34296 CVR52U 25066764 IC50 = 120 nM T34296 C8IBO5 25066765 IC50 = 10 nM T34296 CP85RV 25067176 IC50 = 59 nM T34296 CXP6V8 25067178 IC50 = 1.1 nM T34296 CD2KA4 25102047 IC50 = 4.6 nM T34296 CRW96X 25102048 IC50 = 2.2 nM T34296 CQ3O9P 25102050 IC50 = 0.68 nM T34296 CSHA26 25102051 IC50 = 1.4 nM T34296 C7ADO2 25102197 IC50 = 0.25 nM T34296 CX6D9J 25138245 Ki = 700 nM T34296 C7A6JQ 25138250 Ki = 2000 nM T34296 CR35QP 25144971 IC50 < 25 nM T34296 C0Y5BC 25145683 IC50 < 25 nM T34296 CB7V8Y 25147773 IC50 = 0.12 nM T34296 CEP9Q2 25180867 IC50 = 0.33 nM T34296 C7EH0J 25181615 Ki = 0.3 nM T34296 C6EWF1 25183622 Ki = 1.5 nM T34296 CAH7T2 25183623 Ki = 4.2 nM T34296 CXG2S6 25183625 Ki = 5.8 nM T34296 CHR2P1 25183768 Ki = 4.4 nM T34296 C8IM5D 25263230 IC50 = 120 nM T34296 C7PTR2 25263231 IC50 = 34000 nM T34296 C9MR1P 25263232 IC50 = 670 nM T34296 CW9MK2 25263233 IC50 = 600 nM T34296 CX9L6V 25263234 IC50 = 25446 nM T34296 CJE4M1 25263235 IC50 > 25000 nM T34296 CJ1H5A 25263236 IC50 = 100 nM T34296 C2CGD1 25263237 IC50 = 10 nM T34296 C57UXR 25263238 IC50 = 220 nM T34296 CO4K7N 25263239 IC50 = 2.1 nM T34296 C3TGE2 25263240 IC50 = 3.3 nM T34296 C06WRU 25263241 IC50 = 505 nM T34296 C95AVW 25263242 IC50 = 97 nM T34296 CXT42G 25263243 IC50 = 361 nM T34296 C50DHY 25263244 IC50 = 2500 nM T34296 C6R7SI 25263245 IC50 = 25000 nM T34296 C0H3RD 42627769 IC50 = 1810 nM T34296 CPO1Z3 44123600 Ki = 0.19 nM T34296 CWS64Q 44143474 IC50 = 8624 nM T34296 C7HV5Q 44143475 IC50 = 1900 nM T34296 C06IJY 44143476 IC50 = 440 nM T34296 CVM82U 44143477 IC50 = 415 nM T34296 C5XEB8 44143478 IC50 = 204 nM T34296 CJQF59 44143479 IC50 = 105 nM T34296 C0ZW7S 44143480 IC50 = 349 nM T34296 C7K0YS 44143481 IC50 = 1110 nM T34296 CWU1K0 44143482 IC50 = 835 nM T34296 CA29EQ 44143483 IC50 = 57 nM T34296 CA5P3E 44143484 IC50 = 1451 nM T34296 C7ER1N 44143485 IC50 = 266 nM T34296 C8YNO3 44143486 IC50 = 80 nM T34296 CLJG93 44143487 IC50 = 393 nM T34296 CJB54F 44143488 IC50 = 926 nM T34296 C9LF6X 44143582 IC50 = 0.3 nM T34296 CIH43B 44143583 IC50 = 11 nM T34296 CRO9K7 44143584 IC50 = 0.75 nM T34296 CNT3R8 44143585 IC50 = 6.8 nM T34296 C9TXG7 44143586 IC50 = 1058 nM T34296 CYW27E 44143587 IC50 = 575 nM T34296 C7XOT1 44143588 IC50 = 90 nM T34296 CQ2RN8 44143589 IC50 = 18 nM T34296 CF40SE 44143590 IC50 = 50 nM T34296 CIDW75 44143591 IC50 = 1325 nM T34296 CS7M0P 44143592 IC50 = 145 nM T34296 CKL4T2 44143593 IC50 = 9 nM T34296 CA25DI 44143594 IC50 = 0.7 nM T34296 CW95HZ 44143595 IC50 = 48 nM T34296 CCH26N 44143596 IC50 = 0.5 nM T34296 C6LM5N 44143597 IC50 = 61.5 nM T34296 C9QME0 44143598 IC50 = 9000 nM T34296 CI8Y0R 44143599 IC50 = 197 nM T34296 CE7X2W 44143600 IC50 = 1.3 nM T34296 CYJ0Z4 44143601 IC50 = 12.1 nM T34296 CP1UO5 44143602 IC50 = 300 nM T34296 CP8L7N 44143603 IC50 = 0.6 nM T34296 C6MSK3 44143604 IC50 = 1800 nM T34296 CRL6C0 44143605 IC50 = 0.8 nM T34296 C09OTR 44143606 IC50 = 390 nM T34296 CTM85Q 44143607 IC50 = 25 nM T34296 CV8BO6 44143608 IC50 = 1.3 nM T34296 C8HR2I 44143609 IC50 = 3.9 nM T34296 C90ISP 44143610 IC50 = 3.5 nM T34296 C2J5IT 44143611 IC50 = 2 nM T34296 CO9N4R 44143612 IC50 = 1 nM T34296 C85DBI 44143613 IC50 = 0.8 nM T34296 CQZ2W1 44143614 IC50 = 105 nM T34296 CAP7M2 44143615 IC50 = 60 nM T34296 C3DX9H 44143616 IC50 = 0.9 nM T34296 CIY4K3 44143617 IC50 = 0.6 nM T34296 CRQ0T5 44143618 IC50 = 0.5 nM T34296 COP5G1 44143619 IC50 = 0.4 nM T34296 CM45NB 44143620 IC50 = 110 nM T34296 C20COZ 44143621 IC50 = 1.6 nM T34296 CZC0U7 44143622 IC50 = 13.5 nM T34296 CR4ZF1 44143623 IC50 = 2.8 nM T34296 CZU83Q 44143624 IC50 = 16 nM T34296 CS26DC 44143625 IC50 = 8 nM T34296 C8B3VE 44143626 IC50 = 3.6 nM T34296 CG78RF 44143627 IC50 = 0.9 nM T34296 C8VQS4 44143628 IC50 = 1.7 nM T34296 CKV3C6 44143629 IC50 = 1.4 nM T34296 CK21NW 44143630 IC50 = 1.2 nM T34296 C4ELQ8 44143631 IC50 = 0.7 nM T34296 C9S8YH 44143632 IC50 = 0.7 nM T34296 CCZP24 44143633 IC50 = 230 nM T34296 C3VBX4 44143634 IC50 = 4 nM T34296 CU02HY 44143635 IC50 = 280 nM T34296 C16VZT 44143636 IC50 = 6.9 nM T34296 CSQ0V9 44143637 IC50 = 123 nM T34296 C27UYE 44143638 IC50 = 7.6 nM T34296 C5K2OM 44143639 IC50 = 188 nM T34296 CI7H6E 44143640 IC50 = 49 nM T34296 CH1IR0 44144307 IC50 = 43550 nM T34296 CEC98Q 44182306 IC50 = 430 nM T34296 C6CPZ7 44182307 IC50 = 620 nM T34296 CT80ED 44219901 Ki = 8.2 nM T34296 C94JVY 44219902 IC50 = 41 nM T34296 C7J6GH 44219903 IC50 = 63 nM T34296 C9J7WL 44219904 IC50 = 260 nM T34296 CRQ71E 44219905 IC50 = 600 nM T34296 C4Z0ID 44219906 IC50 = 91 nM T34296 CRNA25 44220092 IC50 = 25 nM T34296 C9T5ZF 44220093 IC50 = 1.4 nM T34296 CV38TE 44222825 IC50 = 15 nM T34296 CJI73R 44222826 IC50 = 7.2 nM T34296 CGQ30N 44222827 Ki = 5.8 nM T34296 CCI64J 44224245 IC50 = 106 nM T34296 C4P2GX 44236892 IC50 = 63 nM T34296 C9RD3F 44236893 IC50 = 57 nM T34296 CTMW04 44236894 IC50 = 31 nM T34296 C7U2CY 44236895 IC50 = 180 nM T34296 C84HYM 44236896 IC50 = 88 nM T34296 C1KY4B 44236897 IC50 = 17 nM T34296 C4PO8V 44236898 IC50 = 245 nM T34296 C8IJ2C 44236899 IC50 = 1550 nM T34296 CG52XV 44236900 IC50 = 6000 nM T34296 C72XPC 44236901 IC50 = 460 nM T34296 C4TDM2 44236902 IC50 = 480 nM T34296 CJW1A3 44236903 IC50 = 290 nM T34296 C9DNJ0 44236904 IC50 > 50000 nM T34296 CW1AF0 44236905 IC50 = 220 nM T34296 CDM1X4 44236906 IC50 = 32 nM T34296 C81SZN 44236907 IC50 = 6 nM T34296 CQ1YS7 44236908 IC50 = 40 nM T34296 C0B2LG 44236909 IC50 = 6 nM T34296 CDI34Y 44236910 IC50 = 25 nM T34296 C6MQO3 44236911 IC50 = 2 nM T34296 C0OY8X 44236912 IC50 = 4 nM T34296 CLRT69 44247751 IC50 = 4.1 nM T34296 CX4VZ8 44248449 IC50 = 40 nM T34296 C3JP6F 44248450 IC50 = 225 nM T34296 CD94XA 44248451 IC50 > 1000 nM T34296 C90ZLT 44248570 IC50 = 187 nM T34296 CF8G2N 44248571 IC50 = 269 nM T34296 CSY0M2 44248572 IC50 = 140 nM T34296 CHM1D7 44248573 IC50 = 1093 nM T34296 CM3Y8J 44248697 IC50 > 1000 nM T34296 CCXS75 44248811 IC50 = 370 nM T34296 CUSR91 44248815 IC50 = 215 nM T34296 COU3Y8 44266817 IC50 = 81.28 nM T34296 CUA5E0 44266818 IC50 = 33 nM T34296 CG23BI 44266830 IC50 = 14.13 nM T34296 CTX92S 44272249 IC50 = 416 nM T34296 CG92WS 44272353 IC50 = 252 nM T34296 CO2Z6K 44272475 IC50 = 5 nM T34296 C63KSL 44272540 IC50 = 47 nM T34296 C20JLP 44272837 IC50 = 123 nM T34296 C4YM6S 44272911 IC50 = 214 nM T34296 C6ON3U 44273235 IC50 = 1590 nM T34296 CSJ50I 44275605 IC50 = 1600 nM T34296 C8CB4A 44275752 IC50 = 14 nM T34296 CVI56W 44275768 IC50 = 300 nM T34296 CV3IQ8 44275769 IC50 = 180 nM T34296 C1O4TU 44275790 IC50 = 2000 nM T34296 CV2WC5 44275791 IC50 = 1600 nM T34296 CUD36E 44275806 IC50 = 110 nM T34296 CPXV83 44275825 IC50 = 1100 nM T34296 CZK8S5 44275954 IC50 = 30 nM T34296 CIK26Z 44276134 IC50 > 3000 nM T34296 C6S3GN 44283598 IC50 = 5 nM T34296 CXE73H 44283613 IC50 = 3 nM T34296 CP3L2U 44283938 IC50 = 170 nM T34296 CET62P 44287169 IC50 > 30000 nM T34296 CJG20R 44287181 IC50 = 6100 nM T34296 CHNI65 44287384 IC50 >> 30000 nM T34296 CB72PO 44287385 IC50 = 27000 nM T34296 C5CT4M 44287386 IC50 = 5100 nM T34296 CS4Z7D 44287398 IC50 = 12000 nM T34296 CF1QK7 44287413 IC50 > 30000 nM T34296 CJ7VW3 44291166 IC50 = 12 nM T34296 C51TQK 44291531 IC50 = 3.8 nM T34296 CF21CS 44291532 IC50 = 3 nM T34296 CU75TB 44291559 IC50 = 96 nM T34296 C06JAO 44291626 IC50 = 20 nM T34296 C2Y0PK 44302023 IC50 = 21 nM T34296 C5S3UO 44302024 IC50 = 11 nM T34296 C8ERW6 44302042 IC50 = 11 nM T34296 CFQ68V 44302071 IC50 = 37 nM T34296 CWB83G 44302076 IC50 = 7 nM T34296 CY1J9U 44302096 IC50 = 17 nM T34296 C5TF4K 44302162 IC50 = 13 nM T34296 CW94ZQ 44302164 IC50 = 200 nM T34296 C5X1WY 44302183 IC50 = 21 nM T34296 C7G3BN 44302200 IC50 = 36 nM T34296 CZP20C 44302339 IC50 = 22 nM T34296 CO73BW 44302357 IC50 = 13 nM T34296 CPC25G 44302409 IC50 = 54 nM T34296 C4NDA2 44302416 IC50 = 26 nM T34296 C24ZWF 44302429 IC50 = 29 nM T34296 C5H6OV 44302627 IC50 = 43 nM T34296 C6QR7C 44302634 IC50 = 67 nM T34296 CG8KJ0 44302661 IC50 = 8 nM T34296 CX1M3Q 44302666 IC50 = 16 nM T34296 CBQ7P3 44302751 IC50 = 21 nM T34296 C36CQP 44302952 IC50 = 32 nM T34296 C4SJF3 44309329 IC50 = 1 nM T34296 C7ED1H 44309330 IC50 = 2 nM T34296 C1E3KF 44309437 IC50 = 4 nM T34296 CH3SU2 44309482 IC50 = 1752 nM T34296 C6N5SL 44309531 IC50 = 18 nM T34296 CO7TS8 44309532 IC50 = 38 nM T34296 CQ7Z0W 44309533 IC50 = 163 nM T34296 CJ0L4P 44309550 IC50 = 3 nM T34296 C6J3WN 44309662 IC50 = 3 nM T34296 CY96UH 44309686 IC50 = 6 nM T34296 C49MHR 44309863 IC50 = 661 nM T34296 CMW0U4 44309879 IC50 = 39 nM T34296 CK6BT0 44309901 IC50 = 142 nM T34296 C5WZR7 44309939 IC50 = 44 nM T34296 C2BLO9 44314811 IC50 = 13 nM T34296 CSY5R3 44314812 IC50 = 17 nM T34296 C0BJ7X 44314813 IC50 = 54 nM T34296 C1V9FZ 44315040 IC50 = 19 nM T34296 C02YGK 44315041 IC50 > 300 nM T34296 C64MTA 44315075 IC50 = 7.7 nM T34296 C85WJB 44315076 IC50 = 9.4 nM T34296 CXLD02 44315105 IC50 = 43 nM T34296 CIJ8H3 44315114 IC50 = 37 nM T34296 C5G7OS 44315115 IC50 = 24 nM T34296 CBP7S0 44315139 IC50 = 44 nM T34296 C4GR1C 44315140 IC50 = 58 nM T34296 CWS3E8 44315141 IC50 = 18 nM T34296 CPAT25 44315142 IC50 = 7.7 nM T34296 C9YK1H 44315143 IC50 = 30 nM T34296 CH48TD 44315155 IC50 = 210 nM T34296 C3VB1J 44315156 IC50 = 31 nM T34296 C79QEK 44315157 IC50 = 11 nM T34296 C62FXJ 44315244 IC50 = 8.3 nM T34296 CB0VI3 44315245 IC50 = 4.3 nM T34296 C4BWR2 44315286 IC50 = 70 nM T34296 CH4YI9 44315311 IC50 = 13 nM T34296 COVF49 44315312 IC50 = 10 nM T34296 C50IQE 44315333 IC50 = 7 nM T34296 C1LC5H 44315334 IC50 = 29 nM T34296 CKAL69 44315860 IC50 = 2 nM T34296 C0HR5Q 44316157 IC50 = 3.981 nM T34296 C5RJ6F 44316310 IC50 = 6 nM T34296 CSA5P7 44316333 IC50 = 1 nM T34296 CS5V0J 44316334 IC50 = 531 nM T34296 CS7D5E 44317086 IC50 = 5 nM T34296 CH70XB 44317451 IC50 = 233 nM T34296 C89IQW 44318090 IC50 = 3 nM T34296 C15WQO 44323336 IC50 = 2.2 nM T34296 C9UOW2 44323407 IC50 = 65 nM T34296 C4C1WD 44323426 IC50 = 4.6 nM T34296 C85JGD 44323430 IC50 = 45.71 nM T34296 CKP12T 44323431 IC50 = 10.4 nM T34296 C4R8OD 44323432 IC50 = 17 nM T34296 COQ6U7 44323456 IC50 = 5.1 nM T34296 CL07GT 44323526 IC50 = 26 nM T34296 CZRF63 44323527 IC50 = 16 nM T34296 CT9M4F 44323539 IC50 = 10.96 nM T34296 CQG24X 44323540 IC50 = 6.2 nM T34296 CND4Y1 44323633 IC50 = 89.13 nM T34296 CBN51C 44324159 IC50 = 87.1 nM T34296 CT01XC 44324546 IC50 = 400 nM T34296 CK5F4S 44324646 IC50 = 400 nM T34296 C6BJ7X 44324656 IC50 = 800 nM T34296 CE6VR2 44324878 IC50 = 400 nM T34296 CYLN13 44324879 IC50 = 2900 nM T34296 CBI48M 44324889 IC50 = 300 nM T34296 CEQ43S 44324934 IC50 = 4000 nM T34296 CRM0C1 44325233 IC50 = 2000 nM T34296 CN0GX1 44325234 IC50 = 200 nM T34296 C5STC3 44325248 IC50 = 300 nM T34296 C2ZH0F 44327181 IC50 = 195 nM T34296 C8V3AO 44327386 IC50 = 41 nM T34296 C0UC5H 44327407 IC50 = 18 nM T34296 C6TPB1 44327409 IC50 = 8 nM T34296 C8ZI0P 44327432 IC50 = 146 nM T34296 CVJ9Q6 44327443 IC50 = 28 nM T34296 C4R9WM 44327681 IC50 = 27 nM T34296 CR40TV 44327695 IC50 = 207 nM T34296 C6IM7G 44327755 IC50 = 28 nM T34296 CHU2P7 44328876 IC50 = 2 nM T34296 C0KA4S 44328937 IC50 = 3 nM T34296 CLT8B6 44328971 IC50 = 4 nM T34296 C7J0ZI 44329016 IC50 = 2 nM T34296 CW24VN 44329040 IC50 = 2 nM T34296 C9J0VO 44329253 IC50 = 2 nM T34296 C90CHA 44329405 IC50 = 600 nM T34296 CB0G1H 44329644 IC50 = 2000 nM T34296 CK9HO7 44329673 IC50 = 100 nM T34296 C07GRS 44329693 IC50 = 19.95 nM T34296 CBH16R 44329694 IC50 = 39.81 nM T34296 CG3E7A 44329712 IC50 = 8 nM T34296 C9SN6I 44329713 IC50 = 199.53 nM T34296 CZ2FW6 44329725 IC50 = 100 nM T34296 CDKI48 44329741 IC50 = 39.81 nM T34296 CK3M2H 44329742 IC50 = 200 nM T34296 C39RDS 44329886 IC50 = 7.943 nM T34296 C3YAF6 44329898 IC50 = 7000 nM T34296 C63RHP 44329909 IC50 = 20 nM T34296 CVQA75 44329910 IC50 = 79.43 nM T34296 C84SLI 44329926 IC50 = 10 nM T34296 CJS6B1 44329927 IC50 = 40 nM T34296 C9R1ZE 44330132 IC50 = 25000 nM T34296 CLU8I7 44330135 IC50 = 3300 nM T34296 C1IE0S 44330147 IC50 = 40000 nM T34296 CPG7N2 44330149 IC50 = 3300 nM T34296 CYP6S4 44330152 IC50 = 5000 nM T34296 CMGA28 44330163 IC50 = 22000 nM T34296 CD0L6S 44331932 IC50 = 3 nM T34296 CHIG68 44331976 IC50 = 6 nM T34296 CF4JN0 44331983 IC50 = 3 nM T34296 CG2AH4 44331984 IC50 = 4 nM T34296 CPB96A 44332003 IC50 = 6 nM T34296 C6RE3I 44332107 IC50 = 0.7 nM T34296 C3L1HQ 44332161 IC50 = 6 nM T34296 CG2Q8W 44332306 IC50 = 84 nM T34296 CY0MQ9 44332313 IC50 = 7 nM T34296 CFP3X8 44334949 IC50 = 96 nM T34296 CV5RF0 44334963 IC50 = 519 nM T34296 C4AOZ7 44334981 IC50 = 218 nM T34296 CXW59C 44334982 IC50 = 22.3 nM T34296 CCH1W8 44334983 IC50 = 3.7 nM T34296 CQ0UI1 44335017 IC50 = 44.2 nM T34296 CX58SB 44335240 IC50 = 5.5 nM T34296 CA96JG 44335285 IC50 = 17 nM T34296 C0Y2CZ 44339375 IC50 = 17 nM T34296 CP12TJ 44339394 IC50 = 4 nM T34296 COR15M 44339402 IC50 = 11 nM T34296 CU5NI2 44339444 IC50 = 6 nM T34296 CISO73 44339448 IC50 = 8 nM T34296 C4QKI6 44339451 IC50 = 7 nM T34296 CEUP59 44339452 IC50 = 4 nM T34296 CU7DZ9 44339462 IC50 = 98 nM T34296 CLT8C6 44339543 IC50 = 3 nM T34296 C6M4UR 44339544 IC50 = 127 nM T34296 C5PQ1B 44339569 IC50 = 7 nM T34296 CA65PF 44339570 IC50 = 20 nM T34296 C4W8LS 44339571 IC50 = 19 nM T34296 COUE24 44339575 IC50 = 40 nM T34296 CMA2L3 44339647 IC50 = 4 nM T34296 CE3MT4 44341611 Ki = 4700 nM T34296 CJTZ45 44341652 Ki = 200000 nM T34296 CE0PL2 44341937 IC50 = 2 nM T34296 C2S1GO 44341947 IC50 = 1.5 nM T34296 C5FG4N 44341974 IC50 = 4.6 nM T34296 CN4UP5 44341977 IC50 = 14 nM T34296 C2S7PL 44341987 IC50 = 0.97 nM T34296 C6EY7C 44342019 IC50 = 24 nM T34296 CK4WL8 44342020 IC50 = 19 nM T34296 C8WH0C 44342056 IC50 = 0.93 nM T34296 CT68XS 44342103 IC50 = 13 nM T34296 CWYV36 44342115 IC50 = 9.7 nM T34296 CER9M5 44342120 IC50 = 0.93 nM T34296 C0KO4U 44342125 IC50 = 0.87 nM T34296 CA1X5L 44342131 IC50 = 49 nM T34296 CIS5M3 44342135 IC50 = 4.6 nM T34296 C80EKJ 44342143 IC50 = 5 nM T34296 C29IPJ 44342160 IC50 = 1.3 nM T34296 CVNF08 44342224 IC50 = 1.5 nM T34296 C5PAS4 44342236 IC50 = 210 nM T34296 CMI0T2 44342251 IC50 = 1.7 nM T34296 CAN54Y 44342308 IC50 = 25 nM T34296 CR9G4Y 44342410 IC50 = 0.56 nM T34296 CD3Y9N 44342428 IC50 = 0.65 nM T34296 CTQ6P4 44344631 IC50 = 2300 nM T34296 CCF94Z 44349787 IC50 = 3.1 nM T34296 C1L2GF 44350073 IC50 = 133 nM T34296 CQ5RN6 44350101 IC50 = 682 nM T34296 CE2X3Q 44350116 IC50 > 100 nM T34296 CQ60YD 44360219 IC50 = 2.1 nM T34296 CT4C6P 44360260 IC50 = 4 nM T34296 CY5I3O 44360286 IC50 = 7.5 nM T34296 C40OCB 44360287 IC50 = 1.4 nM T34296 C90CYD 44367175 IC50 = 3 nM T34296 C2DV0R 44367276 IC50 = 0.4 nM T34296 C5BAW2 44367284 IC50 < 0.4 nM T34296 C2YG5E 44367285 IC50 = 8 nM T34296 CUDF82 44367309 IC50 = 2 nM T34296 CI0ZD9 44371783 IC50 = 176 nM T34296 C4VR5M 44371799 IC50 = 338 nM T34296 C4FHG7 44371800 IC50 = 131 nM T34296 CZ5I8B 44386229 IC50 = 475 nM T34296 C0S7EU 44389231 IC50 = 2500 nM T34296 CN8F1Q 44389253 IC50 > 1200 nM T34296 CB71LT 44389285 IC50 = 270 nM T34296 CZ6PU7 44389401 Ki = 0.33 nM T34296 C40BHI 44389462 Ki = 54 nM T34296 CO7P6Y 44389492 Ki = 5.8 nM T34296 CS1N5F 44389516 Ki = 25 nM T34296 CX25WY 44389537 Ki = 934 nM T34296 CB1RD0 44389551 Ki = 1100 nM T34296 CO4W0Y 44389552 Ki = 0.95 nM T34296 C3YPG6 44390245 IC50 = 8 nM T34296 COG80H 44390258 IC50 = 307 nM T34296 C0U3XR 44390274 IC50 = 363 nM T34296 CAC3F2 44390281 IC50 = 225 nM T34296 CRE9G2 44390289 IC50 = 11 nM T34296 CN41JE 44390299 IC50 = 19.95 nM T34296 C5VBL2 44390300 IC50 = 8.913 nM T34296 C4YUK7 44390304 IC50 = 88 nM T34296 C47EZV 44390314 IC50 = 446 nM T34296 CF65OK 44390317 IC50 = 30.9 nM T34296 CV45JT 44390322 IC50 = 180 nM T34296 C3GU1Q 44390323 IC50 = 52 nM T34296 CAZ2B4 44390326 IC50 = 1063 nM T34296 C2Y7MR 44390338 IC50 = 395 nM T34296 CA47CR 44390351 IC50 = 128 nM T34296 CYW89M 44390352 IC50 = 140 nM T34296 CPK9Z6 44390355 IC50 = 311 nM T34296 CEJH75 44390356 IC50 = 17 nM T34296 CWYM93 44390391 IC50 = 142 nM T34296 C3EZ0W 44391336 IC50 = 19 nM T34296 C1E5JC 44391341 IC50 = 0.54 nM T34296 CT5Y1X 44391344 IC50 = 19 nM T34296 CP0QS3 44391345 IC50 = 4.1 nM T34296 CR0Y3D 44391350 IC50 = 3.1 nM T34296 CMTB94 44391351 IC50 = 3.1 nM T34296 CC7QW9 44391352 IC50 = 1 nM T34296 C0FC5U 44391354 IC50 = 0.61 nM T34296 CMS1Z6 44391356 IC50 = 1.4 nM T34296 CA3NH7 44391357 IC50 = 6 nM T34296 CTK65L 44391360 IC50 = 8 nM T34296 C0S4YB 44391365 IC50 = 53 nM T34296 CN4GJ0 44391366 IC50 = 56 nM T34296 CKL09S 44391376 IC50 = 150 nM T34296 CVTB31 44391377 IC50 > 300 nM T34296 C2R8AW 44391389 IC50 = 390 nM T34296 C3BPI8 44391397 IC50 = 2.1 nM T34296 CW90KP 44391398 IC50 = 1.4 nM T34296 C1N8KB 44391410 IC50 = 18 nM T34296 CB0HI5 44391419 IC50 = 0.87 nM T34296 C5XSH0 44391424 IC50 = 140 nM T34296 CFH41S 44391425 IC50 = 0.95 nM T34296 C49DCW 44391434 IC50 = 9.2 nM T34296 CZ89IE 44391435 IC50 = 5.9 nM T34296 CP0AU9 44391440 IC50 = 3.8 nM T34296 C9BMR7 44391444 IC50 = 0.87 nM T34296 CR4U6B 44391445 IC50 = 3.1 nM T34296 CH59GY 44391449 IC50 = 5 nM T34296 CU7N6G 44391450 IC50 = 3.6 nM T34296 CD5TX3 44391460 IC50 = 190 nM T34296 CCK39J 44391461 IC50 = 3.1 nM T34296 C3V1PB 44391476 IC50 = 1.7 nM T34296 C37DHM 44391486 IC50 = 28 nM T34296 CMGB67 44393214 IC50 = 20 nM T34296 CA1S5T 44393217 IC50 = 21 nM T34296 CSC6N1 44393218 IC50 = 53 nM T34296 CBO9E6 44393239 IC50 = 33 nM T34296 CQNR83 44393261 IC50 = 47 nM T34296 CT1LM8 44393266 IC50 = 17 nM T34296 C0SGF6 44393279 IC50 = 17 nM T34296 CYFC07 44393295 IC50 = 67 nM T34296 C24INM 44393328 IC50 = 32 nM T34296 C15IZJ 44393358 IC50 = 12 nM T34296 C3HP5Q 44393383 IC50 = 19 nM T34296 CS06PD 44393394 IC50 = 42 nM T34296 CFA83O 44393414 IC50 = 97 nM T34296 CCO3S9 44393444 Ki = 1758 nM T34296 CNO4P6 44393516 Ki = 377 nM T34296 C5OIK4 44393520 Ki > 5000 nM T34296 CDG2K7 44393747 IC50 = 1 nM T34296 CWUV21 44393760 IC50 = 140 nM T34296 CQ6WZ5 44393836 IC50 = 5 nM T34296 CR58XA 44393837 IC50 = 1.3 nM T34296 CIH8T9 44393838 IC50 = 28 nM T34296 CK95WI 44393841 IC50 = 46 nM T34296 CAC72Q 44393867 IC50 = 38 nM T34296 CFR4G2 44393892 IC50 = 0.43 nM T34296 CMBJ97 44393897 IC50 = 0.39 nM T34296 CF3M5K 44393910 IC50 = 13 nM T34296 C4YJI9 44393913 IC50 = 300 nM T34296 C0E8BQ 44393936 IC50 = 17 nM T34296 CGU63Q 44393964 IC50 > 300 nM T34296 C8P0IG 44393980 IC50 = 15 nM T34296 CP24NE 44394027 IC50 = 9.8 nM T34296 CHP81Z 44394038 IC50 = 1.1 nM T34296 CKB7S1 44394067 IC50 > 300 nM T34296 CZB81D 44395506 IC50 = 1 nM T34296 CKV57D 44399071 IC50 = 2.8 nM T34296 C0NSO4 44399233 IC50 = 2.1 nM T34296 CRL5D0 44399252 IC50 = 14 nM T34296 CHL9S2 44399294 Ki > 5020 nM T34296 CD49UI 44399312 Ki = 4020 nM T34296 C7IDB0 44399341 IC50 = 3.5 nM T34296 C2UDW8 44399397 IC50 = 7.8 nM T34296 CA0DV5 44399432 IC50 = 1.2 nM T34296 C95RKA 44399451 IC50 = 188 nM T34296 CIA8T3 44399555 Ki > 5020 nM T34296 CV2CQ0 44399635 IC50 = 6.5 nM T34296 CJWB10 44399637 IC50 = 19 nM T34296 CW83LM 44399638 IC50 = 0.5 nM T34296 C7XCI6 44399665 IC50 = 53 nM T34296 CW9MD1 44399704 IC50 = 36 nM T34296 C2JMC1 44399712 IC50 = 4.3 nM T34296 CD8Q2Y 44399731 IC50 = 8 nM T34296 CC16YQ 44399733 IC50 = 1.4 nM T34296 C9KGL0 44404474 IC50 = 0.61 nM T34296 C92KDG 44404475 IC50 = 0.4 nM T34296 C07CGB 44404477 IC50 = 9.5 nM T34296 C7VH3G 44404484 IC50 = 5.9 nM T34296 CC29XL 44404490 IC50 = 55 nM T34296 CCN16G 44404500 IC50 = 17 nM T34296 C69GZU 44404501 IC50 = 3.4 nM T34296 CY6WL5 44404502 IC50 = 1.9 nM T34296 CWGQ46 44404503 IC50 = 4.9 nM T34296 CLXM58 44404504 IC50 = 3.8 nM T34296 C1F9HO 44404506 IC50 = 67 nM T34296 CLU41O 44404507 IC50 = 27 nM T34296 C30DKN 44404553 IC50 = 0.1 nM T34296 C7Z0OH 44404761 IC50 = 83 nM T34296 CIC60V 44406452 IC50 = 4.4 nM T34296 C1F0DR 44406571 IC50 = 20 nM T34296 CT7CD3 44409041 IC50 = 14 nM T34296 CJ2Q8Z 44409042 IC50 = 86 nM T34296 CY3KF2 44409047 IC50 = 17 nM T34296 CT01JW 44409066 IC50 = 4 nM T34296 CJNE37 44409163 IC50 = 2 nM T34296 CVA69I 44409164 IC50 = 4 nM T34296 C9I0JW 44409184 IC50 = 27 nM T34296 C1JSU2 44409197 IC50 = 7 nM T34296 CW4BM3 44409214 IC50 = 8 nM T34296 CVRL76 44409215 IC50 = 2 nM T34296 C9F7HR 44409221 IC50 = 9 nM T34296 CJ70LK 44409222 IC50 = 7 nM T34296 C5J1PS 44409261 IC50 = 1 nM T34296 C06EZF 44409365 IC50 = 7 nM T34296 CV5AW8 44409366 IC50 = 29 nM T34296 C9PS4Q 44409369 IC50 = 24 nM T34296 C1S4GD 44409389 IC50 = 14 nM T34296 C69CGM 44409390 IC50 = 23 nM T34296 C1SKI7 44409405 IC50 = 48 nM T34296 C84ZSL 44411052 Ki = 3 nM T34296 CUE29K 44411053 Ki = 19 nM T34296 C6IKL1 44411602 IC50 = 1.4 nM T34296 CEB0S4 44411823 IC50 = 0.8 nM T34296 CVM7Y3 44413975 IC50 = 24 nM T34296 C4X0GA 44413977 IC50 = 14 nM T34296 CH01EO 44413978 IC50 = 13 nM T34296 CBT0P2 44413982 IC50 = 21 nM T34296 CIJ39D 44413983 IC50 = 39 nM T34296 C9BA0V 44413987 IC50 = 79 nM T34296 CHN85S 44414002 IC50 = 74 nM T34296 C2OJ4B 44414029 IC50 = 177 nM T34296 CF02QK 44419926 IC50 = 1.1 nM T34296 CR1Y6A 44419932 IC50 = 0.85 nM T34296 CVAC97 44419939 IC50 = 3.4 nM T34296 CONP58 44419944 IC50 = 3.9 nM T34296 CYA7G4 44419949 IC50 = 0.4 nM T34296 CNA02B 44419955 IC50 = 6.1 nM T34296 C0Y8RP 44419959 IC50 = 2.6 nM T34296 C0LI1C 44419992 IC50 = 0.84 nM T34296 C5UB4S 44419996 IC50 = 8 nM T34296 CZ5KM8 44421257 IC50 > 10000 nM T34296 CT5PC9 44422672 IC50 = 3.3 nM T34296 CS9D5U 44422720 IC50 = 1.1 nM T34296 CNWM05 44422723 IC50 = 4.2 nM T34296 C58LAY 44422724 IC50 = 13 nM T34296 CDQU41 44422736 IC50 = 63 nM T34296 CVUB56 44422737 IC50 = 24 nM T34296 CB8G2W 44422743 IC50 = 15 nM T34296 CFX42T 44422744 IC50 = 820 nM T34296 C9EL7F 44422749 IC50 = 480 nM T34296 CK5H7O 44429877 IC50 = 4000 nM T34296 CQL1X9 44429878 IC50 = 238 nM T34296 C1CYV2 44429879 IC50 = 295 nM T34296 C7AXP9 44429880 IC50 = 136 nM T34296 CXOS97 44429881 IC50 = 72 nM T34296 C2MQ0I 44429882 IC50 = 43 nM T34296 CQ5PT8 44429883 IC50 = 130 nM T34296 CQRO36 44429884 IC50 = 1159 nM T34296 CM27YB 44429885 IC50 = 155 nM T34296 C9JH0T 44429886 IC50 = 24.4 nM T34296 CD2B3T 44429887 IC50 = 205 nM T34296 C6V1CO 44429888 IC50 = 2040 nM T34296 CBC6W4 44429889 IC50 = 56 nM T34296 C7A0LF 44429890 IC50 = 166 nM T34296 CS0M3L 44429891 IC50 = 385 nM T34296 CX93QY 44429892 IC50 = 147 nM T34296 C8QKS0 44429894 IC50 = 23 nM T34296 CBS47K 44429896 IC50 = 38 nM T34296 CI7TG1 44429897 IC50 = 229 nM T34296 CLJ48T 44429898 IC50 = 195 nM T34296 C3F9CK 44429899 IC50 = 144 nM T34296 C8PVF7 44429900 IC50 = 117 nM T34296 C6U0TK 44429901 IC50 = 104 nM T34296 CBK9M5 44429902 IC50 = 190 nM T34296 C72YFT 44429903 IC50 = 354 nM T34296 CMO9Q3 44429905 IC50 = 449 nM T34296 C8BHL5 44431844 IC50 > 5000 nM T34296 CR1DN9 44431845 IC50 > 5000 nM T34296 CHFB16 44431846 IC50 > 5000 nM T34296 C0C3ZT 44431847 IC50 > 5000 nM T34296 CS49GV 44431848 IC50 > 5000 nM T34296 C4AVK5 44431849 IC50 > 5000 nM T34296 C5DH4Q 44431850 IC50 > 5000 nM T34296 CLHE45 44431851 IC50 > 5000 nM T34296 CYG29L 44431852 IC50 > 5000 nM T34296 C4OF5L 44431853 IC50 > 5000 nM T34296 CWU7G8 44434565 IC50 = 122 nM T34296 C70MGQ 44440455 Ki > 5025 nM T34296 CDY53F 44440460 Ki > 5025 nM T34296 CTB9P6 44440461 Ki = 392 nM T34296 C63RLK 44440462 Ki > 5025 nM T34296 C23JBO 44440463 Ki > 5025 nM T34296 CT9P3Y 44440464 Ki > 5025 nM T34296 CX32AM 44440465 Ki > 5025 nM T34296 C6FOC7 44440466 Ki > 5025 nM T34296 CMPX37 44440467 Ki > 5025 nM T34296 CV4F6Z 44440468 Ki > 5025 nM T34296 C6K8VB 44440469 Ki > 5025 nM T34296 C4Y0UM 44440470 Ki > 5025 nM T34296 CHU49A 44440471 Ki > 5025 nM T34296 C8OI4L 44440472 Ki > 5025 nM T34296 CV58YW 44441018 Ki > 5025 nM T34296 CV85PN 44441019 Ki > 5025 nM T34296 C5O2WK 44441020 Ki > 5025 nM T34296 CU67WS 44441021 Ki > 5025 nM T34296 CXZ53B 44441022 Ki = 2462 nM T34296 C8S7UT 44441023 Ki > 5025 nM T34296 CT4PZ9 44441024 Ki > 5025 nM T34296 CU9GE6 44441025 Ki > 5025 nM T34296 CB2IT4 44441026 Ki > 5025 nM T34296 CN4X2F 44441027 Ki = 3136 nM T34296 CPF45Y 44441028 Ki > 5025 nM T34296 CAM23N 44441029 Ki > 5025 nM T34296 C23BPG 44441030 Ki > 5025 nM T34296 C5YMT6 44441031 Ki > 5025 nM T34296 C9A6GJ 44441032 Ki > 5025 nM T34296 CYSU19 44441033 Ki > 5025 nM T34296 CB9P0C 44442303 IC50 = 1200 nM T34296 C7HO0Y 44442304 IC50 = 1100 nM T34296 CAR3S2 44442305 IC50 = 1170 nM T34296 CZK0A9 44442306 IC50 = 2860 nM T34296 C71MCV 44442307 IC50 = 1200 nM T34296 CN70HO 44442308 IC50 = 1110 nM T34296 CVE5P0 44442309 IC50 = 840 nM T34296 CGS18B 44442311 IC50 = 1010 nM T34296 CIZL27 44442312 IC50 = 1370 nM T34296 CCFV76 44442313 IC50 = 1190 nM T34296 CZ2PE6 44442315 IC50 = 950 nM T34296 C2N8BW 44442316 IC50 = 1740 nM T34296 CGR6E7 44442318 IC50 > 16666 nM T34296 C97ZHM 44442319 IC50 > 16666 nM T34296 C3DIB8 44442320 IC50 > 16666 nM T34296 C9IQD0 44444485 IC50 = 8.9 nM T34296 C64FGU 44444487 IC50 = 2.9 nM T34296 CR4O1V 44444516 IC50 = 138 nM T34296 CGZ20Y 44444519 IC50 = 7.33 nM T34296 CV4MK5 44444526 IC50 = 12 nM T34296 CI20ZD 44444531 IC50 = 0.6 nM T34296 C91QFR 44444569 IC50 = 0.49 nM T34296 CG3P8M 44444573 IC50 = 0.11 nM T34296 CO46QB 44444576 IC50 = 0.96 nM T34296 C9L4DH 44444578 IC50 = 0.1 nM T34296 CBC28D 44444580 IC50 = 0.4 nM T34296 CV0CI2 44444582 IC50 = 0.08 nM T34296 CL4BX1 44445917 IC50 = 15.85 nM T34296 CKW5G7 44445918 IC50 = 1 nM T34296 CE0O2Z 44445919 IC50 = 20.89 nM T34296 CSKN69 44455242 IC50 = 4 nM T34296 C3J1SV 44455676 IC50 = 11 nM T34296 C38VBL 44455836 IC50 = 13.4 nM T34296 CG0Z7I 44478924 IC50 = 2700 nM T34296 CFO27Y 44478926 IC50 = 84 nM T34296 CBZJ29 44478927 IC50 = 25 nM T34296 CRJ24K 44479197 IC50 = 12 nM T34296 CGOH82 44479198 IC50 = 940 nM T34296 CLV56M 44479199 IC50 = 78 nM T34296 CY92OQ 44479458 IC50 = 20000 nM T34296 CH1QG9 44479459 IC50 = 260 nM T34296 CB1NT7 44479460 IC50 = 62 nM T34296 C0JQ9L 44479699 IC50 = 74 nM T34296 C0DN1Q 44479700 IC50 = 55000 nM T34296 CTG24W 44479702 IC50 = 1800 nM T34296 CGZ49M 44479703 IC50 = 190 nM T34296 CAK94X 44563337 IC50 = 213 nM T34296 CY1A8V 44564505 IC50 = 3 nM T34296 C47XUD 44571675 IC50 > 200000 nM T34296 CQ7W5I 44580110 Ki > 5000 nM T34296 CWD32S 44580184 IC50 = 2277 nM T34296 CH8QS0 44596287 IC50 = 0.6 nM T34296 CW5A2D 44608129 IC50 = 8 nM T34296 CT7KX5 44608938 IC50 = 33 nM T34296 CJRP30 44608939 IC50 = 26 nM T34296 COI5K3 44608942 IC50 = 28 nM T34296 CS4C5T 44609098 IC50 = 2 nM T34296 CMLV87 44609099 IC50 = 28 nM T34296 C3T9SV 44609100 IC50 = 2.9 nM T34296 C0KR6J 44626353 IC50 = 1130 nM T34296 C25QLI 44626354 IC50 = 3760 nM T34296 CA1YC9 44626604 Ki = 19 nM T34296 CK6S5H 44626708 Ki = 1200 nM T34296 C0EJ1F 44626709 Ki = 30 nM T34296 CZR23J 44626710 Ki > 10000 nM T34296 CQB06H 44626711 Ki = 24 nM T34296 C19LWR 44634267 IC50 = 0.58 nM T34296 CZP79X 45268488 IC50 = 6.1 nM T34296 CK50JB 45268522 IC50 = 35 nM T34296 C2B0GI 45268787 Ki = 1.5 nM T34296 CVG5I2 45269378 IC50 = 11 nM T34296 CQC5Y4 45269386 IC50 = 14 nM T34296 CACH13 45269631 IC50 = 9.4 nM T34296 C2HI5Q 45269910 IC50 = 13800 nM T34296 C84JSF 45269911 IC50 = 60000 nM T34296 CTOH60 45270200 IC50 = 7.1 nM T34296 C2H5IY 45271017 IC50 = 7.4 nM T34296 C0YT8W 45271893 IC50 = 4.8 nM T34296 CVNO86 45271894 IC50 = 2.3 nM T34296 C7OQB3 45271912 IC50 = 13 nM T34296 C3SWC7 45272759 IC50 = 40 nM T34296 C36HRP 45377138 IC50 = 14 nM T34296 C6B7ZY 45377564 IC50 = 90 nM T34296 C5HAR6 45377565 IC50 = 150 nM T34296 CZYH47 45377567 IC50 = 56000 nM T34296 CKR0Q8 45377703 IC50 = 120 nM T34296 CMPE63 45482676 IC50 = 7900 nM T34296 CGH1U8 45482997 IC50 = 50200 nM T34296 C8AUI5 45482999 IC50 > 98000 nM T34296 C9W7IP 45483016 IC50 = 26100 nM T34296 CPB42K 45483022 IC50 = 33500 nM T34296 CBG76X 45483023 IC50 = 41900 nM T34296 CDW4C8 45483036 IC50 > 98000 nM T34296 CSX5I9 46175170 IC50 = 3.4 nM T34296 C56WVI 46184724 Ki = 3600 nM T34296 C8A3ER 46207232 IC50 = 2 nM T34296 CNF8R2 46207262 IC50 = 28 nM T34296 CT85VJ 46207292 IC50 = 2 nM T34296 CFW09H 46207358 IC50 = 6 nM T34296 C2W1KN 46225418 Ki = 65.3 nM T34296 CEVP65 46225419 Ki = 75.9 nM T34296 CA9QD6 46225437 Ki = 43.4 nM T34296 C25OWI 46225438 Ki = 36.7 nM T34296 CVL2I0 46225439 Ki = 2.1 nM T34296 CHKW61 46225440 Ki = 227 nM T34296 CTU9S1 46225452 Ki = 18.1 nM T34296 C9L8TO 46225453 Ki = 16.5 nM T34296 CJO87P 46225454 Ki = 22.3 nM T34296 C9KM3H 46225455 Ki = 5.3 nM T34296 CF12SQ 46225473 Ki = 28.6 nM T34296 CD6M3V 46225474 Ki = 3.6 nM T34296 C45RIP 46225475 Ki = 4.4 nM T34296 CW0G8P 46225476 Ki = 0.18 nM T34296 CGK72P 46225491 Ki = 2.5 nM T34296 CW42CR 46225492 Ki = 31.3 nM T34296 CJS16C 46225493 Ki = 4.2 nM T34296 C9WDJ6 46225506 Ki = 22.1 nM T34296 CV0G1O 46225507 Ki = 6.7 nM T34296 CG3SX7 46225508 Ki = 1.5 nM T34296 CP8NT9 46225509 Ki = 0.16 nM T34296 C7S1QD 46225519 Ki = 1.5 nM T34296 CWY81P 46225520 Ki = 7.5 nM T34296 C0ZIX3 46225521 Ki = 1.4 nM T34296 C6LY8C 46225536 Ki = 0.26 nM T34296 CZO14V 46225537 Ki = 0.62 nM T34296 C7HNV9 46225538 Ki = 0.22 nM T34296 CL2U4Z 46829322 Ki = 1 nM T34296 CH0Z1E 46844314 Ki > 40000 nM T34296 C7IXV6 46849757 IC50 > 10000 nM T34296 C20BTY 46856241 Ki = 3300 nM T34296 C5L8GF 46871738 IC50 = 0.6 nM T34296 CR1KF7 46871739 IC50 = 1 nM T34296 C8Q6YR 46871740 IC50 = 0.42 nM T34296 C58YSM 46871741 IC50 = 4 nM T34296 CR96AK 46890762 IC50 = 90 nM T34296 C5G9FX 46890763 IC50 = 6.7 nM T34296 COP78K 46890764 IC50 = 18 nM T34296 C60QSB 46890765 IC50 = 6 nM T34296 CQ5P9V 46890766 IC50 = 6.7 nM T34296 CB90YN 46890767 IC50 = 12.2 nM T34296 CUA7L6 46890821 IC50 = 10.7 nM T34296 C9BNQ7 46890822 IC50 = 6.4 nM T34296 CTF20Y 46890823 IC50 = 30 nM T34296 CR3QW7 46891107 IC50 = 2.7 nM T34296 C5MK3A 46891108 IC50 = 7.7 nM T34296 CQ5E1H 46891109 IC50 = 9 nM T34296 C0NW9D 46891110 IC50 = 130 nM T34296 C91LGI 46891170 IC50 = 8 nM T34296 CGI5B4 46891171 IC50 = 20 nM T34296 CZPM12 46891172 IC50 = 0.63 nM T34296 C2V6MW 46891173 IC50 = 1.9 nM T34296 CZWT45 46891207 IC50 = 28.6 nM T34296 CFE58Q 46891208 IC50 = 3.3 nM T34296 C8S7QX 46891209 IC50 = 2.4 nM T34296 C5Y0MN 46891255 IC50 = 17.5 nM T34296 CJ16SE 46891256 IC50 = 0.7 nM T34296 C7Y9TE 46891257 IC50 = 42.5 nM T34296 C7DT6W 46891258 IC50 = 32.7 nM T34296 CLF7Y4 46891311 IC50 = 28.8 nM T34296 C2IN7Y 46891312 IC50 = 35 nM T34296 CNXU57 46891313 IC50 = 11.3 nM T34296 CJB5D0 46891314 IC50 = 33.7 nM T34296 CVK0E5 46891356 IC50 = 11.4 nM T34296 C89RPO 46891357 IC50 = 7 nM T34296 CVB6K4 46891358 IC50 = 11 nM T34296 C67WEK 46891359 IC50 = 11.4 nM T34296 CPQ37V 46891414 IC50 = 70 nM T34296 C5LTI6 46891459 IC50 = 35 nM T34296 C92FBL 46891460 IC50 = 24.5 nM T34296 C1A0OE 46891522 IC50 = 9 nM T34296 C2I6FV 46891523 IC50 = 6.2 nM T34296 CAZ9Q5 46891524 IC50 = 4.4 nM T34296 CG02KB 46891525 IC50 = 50 nM T34296 C7ZG8J 46891526 IC50 = 18.1 nM T34296 CRQ13J 46891580 IC50 = 50 nM T34296 CERM39 46891581 IC50 = 28 nM T34296 CN8WF9 46891582 IC50 = 45 nM T34296 C86RLM 46891583 IC50 = 25.1 nM T34296 CM7S5T 46891584 IC50 = 40 nM T34296 CRY18A 46891617 IC50 = 26.8 nM T34296 C0S9WB 46919610 Ki = 3500 nM T34296 C6U1ZJ 46934733 IC50 = 24 nM T34296 CX89ON 46935023 IC50 = 11 nM T34296 CJ5U9I 46935024 IC50 = 8 nM T34296 CE3H7I 46938726 IC50 = 0.2 nM T34296 C9T0HR 46938727 IC50 = 0.6 nM T34296 C0YR7M 46938728 IC50 < 0.1 nM T34296 C2S7PK 46942365 Ki = 1.7 nM T34296 C2TE8J 47162079 IC50 = 39000 nM T34296 CE35HQ 49865150 IC50 = 100 nM T34296 C6YF2O 49865151 IC50 = 3300 nM T34296 CW5Q1C 49865207 IC50 = 110 nM T34296 C1FT8V 49865208 IC50 = 140 nM T34296 C0MC4H 49865209 IC50 = 75 nM T34296 CG17QX 49865271 IC50 = 180 nM T34296 CAR87K 49865272 IC50 = 330 nM T34296 CD8NS5 49865273 IC50 = 310 nM T34296 CJ5R6M 49865325 IC50 = 72 nM T34296 C6K2OQ 49865326 IC50 = 140 nM T34296 C8JM0Q 49865327 IC50 = 8 nM T34296 C0FJ1B 49865379 IC50 = 42 nM T34296 CD45PA 49865380 IC50 = 31 nM T34296 CF4VU8 49865381 IC50 = 10 nM T34296 CY1LX7 49865382 IC50 = 4 nM T34296 C16SGP 49865429 IC50 = 9 nM T34296 C6LI1B 49865430 IC50 = 100 nM T34296 C4GOT9 49865431 IC50 = 29 nM T34296 CFS08O 49865432 IC50 = 27 nM T34296 C6QYN3 49865473 IC50 = 3 nM T34296 C8QH3B 49865474 IC50 = 7 nM T34296 CE0M1T 49865521 IC50 = 25 nM T34296 CX67WT 49865522 IC50 = 9 nM T34296 CFRI63 49865523 IC50 = 36 nM T34296 CJR6H7 49865573 IC50 = 5 nM T34296 C7XW1Q 50907084 Ki = 1.7 nM T34296 C8RL5Q 50907292 Ki = 18 nM T34296 CUD7O0 50941549 IC50 > 10000 nM T34296 CX8N4D 50990920 IC50 = 430 nM T34296 CXF4V3 50990921 IC50 > 8100 nM T34296 CU2SX3 51355576 Ki = 7730 nM T34296 CLA96C 53232689 Ki = 0.6 nM T34296 C3BGW0 53233015 Ki > 40000 nM T34296 CZ06OY 53233469 IC50 = 0.66 nM T34296 CMQZ70 53242178 IC50 > 31000 nM T34296 CC9HK5 53245646 IC50 = 79.43 nM T34296 CRI92N 53311230 IC50 = 100 nM T34296 CB09MA 53318910 IC50 = 7.6 nM T34296 C47DIU 53318911 IC50 = 530 nM T34296 CC6DR2 53318912 IC50 = 23000 nM T34296 CWH47R 53319228 Ki = 2.9 nM T34296 C7V1NC 53320225 IC50 = 2300 nM T34296 CVH2B7 53320226 IC50 > 16000 nM T34296 CO8QK2 53320227 IC50 = 350 nM T34296 CNS3F2 53321542 IC50 = 16000 nM T34296 C1N2BX 53322876 IC50 = 2300 nM T34296 CSYW40 53322877 IC50 = 27000 nM T34296 CGUC59 53322878 IC50 = 4600 nM T34296 C3QHA6 53322879 IC50 > 4500 nM T34296 C1VNZ9 53324198 IC50 = 180 nM T34296 C0H7FQ 53324260 IC50 = 6700 nM T34296 CZD9L1 53324788 IC50 = 3800 nM T34296 CU7YG9 53325497 IC50 = 260 nM T34296 C4G1HK 53325498 IC50 = 17000 nM T34296 CO5L1I 53325499 IC50 = 14000 nM T34296 CZA03W 53326760 IC50 = 370 nM T34296 CM53CG 53326761 IC50 = 6100 nM T34296 CWR6T4 53326860 IC50 = 570 nM T34296 C6Y2EV 53374826 IC50 > 100000 nM T34296 CQ04KO 53389286 IC50 = 3 nM T34296 C1IFJ8 53957122 IC50 = 97000 nM T34296 CBL30Y 54181369 IC50 > 10000 nM T34296 CSUW40 54352406 IC50 = 18 nM T34296 C3M8GZ 54580051 IC50 = 46000 nM T34296 CL0WM9 54580052 IC50 > 10000 nM T34296 CK26XF 54580053 IC50 > 10000 nM T34296 CS1LM9 54580054 IC50 = 154 nM T34296 C3LF0P 54580544 Ki = 3.7 nM T34296 CA8U9V 54580837 IC50 = 8 nM T34296 C8PE1G 54581030 IC50 = 570 nM T34296 CVO09J 54581546 Ki = 0.66 nM T34296 CWB2Q6 54581896 IC50 = 1.2 nM T34296 CVK72M 54582073 IC50 = 940 nM T34296 CBK18O 54582074 IC50 > 10000 nM T34296 CP2F1B 54582075 IC50 > 10000 nM T34296 CZNU23 54582076 IC50 > 10000 nM T34296 C0U5HZ 54582077 IC50 > 4100 nM T34296 CSTG96 54582078 IC50 = 1400 nM T34296 C8SG9Y 54582079 IC50 > 10000 nM T34296 CZI6S3 54582080 IC50 = 5900 nM T34296 CD09BZ 54582543 IC50 = 0.7 nM T34296 CH6Q2Z 54583016 IC50 > 10000 nM T34296 C3V9LQ 54583017 IC50 = 260 nM T34296 CT80KQ 54583018 IC50 > 600 nM T34296 CPT4L5 54583019 IC50 = 8400 nM T34296 CK52YD 54583511 Ki = 1.7 nM T34296 CF0SK8 54583712 IC50 = 0.3 nM T34296 CBEV27 54584024 IC50 = 1700 nM T34296 CM87DP 54584025 IC50 = 1100 nM T34296 C28GKQ 54585927 IC50 > 10000 nM T34296 CAZ76E 54586892 IC50 = 4600 nM T34296 CM0OQ3 54586893 IC50 > 10000 nM T34296 CK1NS7 54586894 IC50 > 10000 nM T34296 CMC4Y1 54586895 IC50 > 10000 nM T34296 C2MKX5 54586896 IC50 = 2000 nM T34296 CU91QP 54586897 IC50 > 10000 nM T34296 CI08RQ 54586898 IC50 = 780 nM T34296 C6PRI4 54586899 IC50 > 10000 nM T34296 CG37UX 54587429 Ki = 1.2 nM T34296 CL9SC3 54587769 Ki = 14100 nM T34296 CGH0S7 54589400 IC50 > 100000 nM T34296 C9P5ES 54752445 IC50 = 0.7 nM T34296 C0HKC9 54752446 IC50 = 0.4 nM T34296 CIV16T 56659712 IC50 = 25118.86 nM T34296 C06AWP 56659713 IC50 > 398107.17 nM T34296 CTM86X 56659714 IC50 = 251.19 nM T34296 CFZ48A 56659715 IC50 = 501.19 nM T34296 CC94RE 56663176 IC50 = 3162.28 nM T34296 C5EA4B 56666624 IC50 = 50118.72 nM T34296 CCSY94 56666625 IC50 > 398107.17 nM T34296 C40WKH 56670032 IC50 = 19952.62 nM T34296 C5GOU2 56670033 IC50 = 5011.87 nM T34296 C9MW0X 56670034 IC50 = 125.89 nM T34296 C5FE3V 56673547 IC50 > 398107.17 nM T34296 C4TSJ8 56673548 IC50 = 25118.86 nM T34296 CFLI43 56673549 IC50 > 100000 nM T34296 CADI17 56673550 IC50 > 398107.17 nM T34296 CG0N3B 56673551 IC50 = 398.11 nM T34296 CF98LT 56676871 IC50 = 50118.72 nM T34296 C4EHL2 56676872 IC50 = 316.23 nM T34296 CP98QO 56680187 IC50 = 25118.86 nM T34296 CG8D6A 56680188 IC50 = 63.1 nM T34296 CA8R2T 56680189 IC50 = 2511.89 nM T34296 C62FZC 56835063 IC50 = 1980 nM T34296 CKJ9S1 56835167 IC50 = 9.5 nM T34296 C21CLZ 56835168 IC50 = 52 nM T34296 C0L2TS 56835169 IC50 = 300 nM T34296 CKEV19 56850269 IC50 > 500000 nM T34296 C13DBR 56850270 IC50 > 500000 nM T34296 C05CTJ 56850271 IC50 = 15000 nM T34296 CX8QD5 56850272 IC50 = 82000 nM T34296 C1I9RE 56850407 IC50 = 9600 nM T34296 CVJ90W 56850408 IC50 = 2500 nM T34296 CPI5G0 56850409 IC50 = 2400 nM T34296 CFR3E5 56850410 IC50 > 26000 nM T34296 CRE5O1 56850411 IC50 = 250 nM T34296 CK47BT 56928417 IC50 = 3.5 nM T34296 C8TH2F 56945850 IC50 = 48 nM T34296 CD72TG 56945851 IC50 = 16 nM T34296 C8J4SC 56945854 IC50 = 87 nM T34296 C1AIZ6 56945963 IC50 = 9 nM T34296 CXQC91 56945964 IC50 = 51 nM T34296 CM4H9D 56945965 IC50 = 94 nM T34296 CUT4S2 56946063 IC50 = 605 nM T34296 C2CQR8 56946064 IC50 = 7 nM T34296 C2H8PG 56946065 IC50 = 23 nM T34296 CW2P6A 56946167 IC50 = 21 nM T34296 CT8S3G 56946168 IC50 = 40 nM T34296 C8YID1 56970123 IC50 > 300000 nM T34296 CI5A2O 56970124 IC50 = 5200 nM T34296 CTW18D 56970125 IC50 = 3200 nM T34296 CIK96H 56970340 IC50 = 2600 nM T34296 C1SBD6 56970341 IC50 = 4900 nM T34296 CHA5Q6 56970342 IC50 = 4900 nM T34296 C7A5GT 56970550 IC50 = 5500 nM T34296 C10BMZ 57127110 IC50 > 10000 nM T34296 CQU16V 57339411 Ki = 49 nM T34296 C6LM3B 57339412 Ki = 14 nM T34296 CNVG85 57339413 Ki = 12 nM T34296 C0IU4S 57390230 IC50 = 9.6 nM T34296 CCN3K2 57390233 IC50 = 4300 nM T34296 CJ49DO 57390234 IC50 = 24700 nM T34296 CU34JA 57390237 IC50 = 4000 nM T34296 C9SD5O 57390259 IC50 = 1.4 nM T34296 CI0X9S 57391136 IC50 = 0.6 nM T34296 CD9J1C 57391201 IC50 = 79.43 nM T34296 C6ZAX3 57391202 IC50 = 316.23 nM T34296 C1POE0 57391203 IC50 = 100 nM T34296 CN2H9K 57391204 IC50 = 39.81 nM T34296 CR8MW2 57391205 IC50 = 10 nM T34296 CA25DM 57391224 IC50 = 7 nM T34296 C6P9XK 57391225 IC50 = 18 nM T34296 CJC7M9 57392022 IC50 = 1.1 nM T34296 CAL94F 57392025 IC50 = 2.6 nM T34296 CA6L5W 57392045 IC50 = 2 nM T34296 CH1I4N 57392901 IC50 = 13 nM T34296 C7CV1B 57392902 IC50 = 361 nM T34296 C25FAK 57392903 IC50 = 1.8 nM T34296 C4CK0Q 57392968 IC50 = 79.43 nM T34296 CNQ9B2 57392969 IC50 = 199.53 nM T34296 CU3SG5 57392970 IC50 = 5011.87 nM T34296 C4NYE5 57392971 IC50 = 2511.89 nM T34296 CTYP14 57392972 IC50 = 50.12 nM T34296 C5VB0U 57392973 IC50 = 25.12 nM T34296 CMQL31 57392974 IC50 = 100 nM T34296 C39OHF 57392975 IC50 = 79.43 nM T34296 CX89EL 57392993 IC50 = 32 nM T34296 CB64TD 57393744 IC50 = 5.6 nM T34296 C3CA9G 57393746 IC50 = 0.1 nM T34296 CP5BX6 57394607 IC50 = 3 nM T34296 CA09RY 57394649 IC50 = 10 nM T34296 CDCW73 57394678 IC50 = 220000 nM T34296 CH6BA3 57394709 IC50 = 31.62 nM T34296 CD1CO2 57394710 IC50 = 2511.89 nM T34296 CNOH63 57394711 IC50 = 74 nM T34296 C1CYK9 57394729 IC50 = 15 nM T34296 C9JC3H 57394730 IC50 = 2.2 nM T34296 C80FML 57394731 IC50 = 3.2 nM T34296 CYFJ06 57394732 IC50 = 242 nM T34296 C27AQN 57395458 IC50 = 1.4 nM T34296 C10PRG 57395459 IC50 = 0.7 nM T34296 C42XNM 57395460 IC50 = 4.6 nM T34296 C17DMO 57395461 IC50 = 0.1 nM T34296 CZX7S9 57395466 IC50 = 2.7 nM T34296 CQ4JU6 57395492 IC50 = 12 nM T34296 COXA03 57396390 IC50 = 7 nM T34296 CO17CH 57396398 IC50 = 12 nM T34296 CDES09 57396473 IC50 = 19.95 nM T34296 CONH52 57396474 IC50 = 50.12 nM T34296 CV51ME 57396475 IC50 = 100 nM T34296 C7QD2T 57396476 IC50 = 398.11 nM T34296 CJB27Z 57396489 IC50 = 12 nM T34296 C34RZI 57396490 IC50 = 1 nM T34296 CBY21D 57397314 IC50 = 1.4 nM T34296 CD6Q9F 57398187 IC50 = 180 nM T34296 CSX81J 57398194 IC50 = 165 nM T34296 CBH82N 57398195 IC50 = 0.3 nM T34296 C2INW7 57398264 IC50 > 10000 nM T34296 C0YHM7 57398273 IC50 = 1.3 nM T34296 C5R1PU 57398274 IC50 = 34 nM T34296 CR59KW 57398991 IC50 = 450 nM T34296 C0ZL1D 57399843 IC50 = 100 nM T34296 CI6WB3 57399844 IC50 = 3892 nM T34296 C5SVE2 57399911 IC50 = 316.23 nM T34296 CZ4GX2 57399912 IC50 = 31.62 nM T34296 C4J5LE 57399913 IC50 = 63.1 nM T34296 CH1J9Q 57399914 IC50 = 63.1 nM T34296 CGTF67 57399915 IC50 = 630.96 nM T34296 CI6AZ8 57399916 IC50 = 1584.89 nM T34296 CAKW95 57399917 IC50 > 10000 nM T34296 CD50CO 57399918 IC50 = 50.12 nM T34296 C82HGR 57399936 IC50 = 480 nM T34296 CAX15U 57399937 IC50 = 603 nM T34296 C5U9NO 57400708 IC50 = 1 nM T34296 CBZ36R 57401604 IC50 = 0.05 nM T34296 CM9D3A 57401688 IC50 = 251.19 nM T34296 CF02UP 57401689 IC50 = 12.59 nM T34296 CVO56U 57401690 IC50 = 63.1 nM T34296 CN27EP 57401691 IC50 = 39.81 nM T34296 CJLZ14 57401692 IC50 = 25.12 nM T34296 C2AI8P 57401693 IC50 = 100 nM T34296 CLNT30 57401717 IC50 = 24 nM T34296 CKL68A 57401718 IC50 = 3.6 nM T34296 COP3C5 57402482 IC50 = 7.1 nM T34296 C6HZ1P 57402483 IC50 = 5.2 nM T34296 CGMQ47 57402485 IC50 = 2.2 nM T34296 C37JZN 57402486 IC50 = 1600 nM T34296 CT26AL 57403355 IC50 = 176 nM T34296 C6OQH8 57403420 IC50 = 10 nM T34296 C2Z6EC 57403421 IC50 = 100 nM T34296 CA5Z2V 57403422 IC50 = 50.12 nM T34296 C9O5HA 57403423 IC50 = 1000 nM T34296 CK68EY 57403424 IC50 = 79.43 nM T34296 CQN8L6 57403445 IC50 = 2.2 nM T34296 C2L1SE 57403446 IC50 = 1.3 nM T34296 C2MH8O 57523473 IC50 = 0.09 nM T34296 C57CEM 57523505 IC50 = 1 nM T34296 CS8W4L 57523538 IC50 = 10 nM T34296 CIT7B9 57523539 IC50 = 6 nM T34296 C56QXU 57523540 IC50 = 4 nM T34296 CX8IU3 57523541 IC50 = 18 nM T34296 CE8CL9 57523575 IC50 = 5 nM T34296 CWUP89 57523576 IC50 = 0.006 nM T34296 CT2QS3 57523577 IC50 = 0.02 nM T34296 CK6M0Y 57523578 IC50 = 0.04 nM T34296 C0HVU7 57523611 IC50 = 1 nM T34296 C5Q0ND 57523641 IC50 = 6 nM T34296 CWH7V8 57561293 IC50 = 684 nM T34296 C1PHI6 57708731 IC50 = 0.078 nM T34296 C1MW3I 57708751 IC50 = 0.027 nM T34296 CE27US 57708758 IC50 = 0.026 nM T34296 C2PF5O 57708776 IC50 = 0.043 nM T34296 CF2Z7W 57708783 IC50 = 0.033 nM T34296 C76ABG 57708790 IC50 = 0.1 nM T34296 C9KV2W 57708792 IC50 = 1.5 nM T34296 CE36GP 57708799 IC50 = 0.29 nM T34296 CK6H4D 57708802 IC50 = 0.44 nM T34296 CX5B1P 57708811 IC50 = 0.093 nM T34296 CA3E8P 57708824 IC50 = 0.091 nM T34296 CQ1E7H 57708842 IC50 = 0.059 nM T34296 C23QGY 57708843 IC50 = 4.9 nM T34296 C4NCK5 57708858 IC50 = 0.29 nM T34296 C2J5CW 57708880 IC50 = 2.6 nM T34296 CSO4R8 57708881 IC50 = 0.057 nM T34296 CS25LJ 57708883 IC50 = 0.074 nM T34296 C1K6AP 57708886 IC50 = 0.064 nM T34296 CY1N3J 57792153 IC50 = 1230 nM T34296 CCKD80 58307579 Ki = 28 nM T34296 C1EJ4S 59379730 Ki = 0.59 nM T34296 CK93UZ 59788426 IC50 = 1.3 nM T34296 C8ITK7 59794408 IC50 = 59.1 nM T34296 CSO3W8 59794423 IC50 = 28.9 nM T34296 C6JE9N 59794437 IC50 = 11.5 nM T34296 C7ECU2 59794447 IC50 = 21 nM T34296 C52ESR 66559934 IC50 > 50000 nM T34296 C57ARI 66560021 IC50 > 25000 nM T34296 CU58DB 66560022 IC50 > 25000 nM T34296 C16RDM 66560389 IC50 = 7900 nM T34296 C8RZG9 66560479 IC50 = 7900 nM T34296 C5AQG2 68724898 Ki = 16.6 nM T34296 CC2UE5 68726681 Ki = 0.2 nM T34296 CJU60O 68793626 Ki = 6.3 nM T34296 CMG96N 68794188 Ki = 32.9 nM T34296 C9AL6F 68794211 Ki = 47.2 nM T34296 C7A5PI 68795150 Ki = 21.2 nM T34296 C4IPW3 68795152 Ki = 3.8 nM T34296 CNS46M 68795882 Ki = 29.3 nM T34296 CHL56C 68799256 Ki = 1.4 nM T34296 CT2K3G 70265758 Ki = 2.7 nM T34296 CHRO48 70266605 Ki = 11.7 nM T34296 C34LYX 70266607 Ki = 7.7 nM T34296 COD03W 70267879 Ki = 0.25 nM T34296 CG38ZM 70267887 Ki = 4.5 nM T34296 C3CEL7 70267989 Ki = 23.8 nM T34296 CJHN06 70268164 Ki = 38.5 nM T34296 C50CAL 70268171 Ki = 2.1 nM T34296 CWP71E 70269104 Ki = 16.5 nM T34296 CVWI31 70269555 Ki = 1.2 nM T34296 CGD3B2 70269997 Ki = 5.8 nM T34296 C0GKT8 70685026 IC50 = 3.9 nM T34296 C8B6WD 70688393 IC50 = 18520 nM T34296 CGR3J2 70688394 IC50 = 13170 nM T34296 CFM0Q5 70690777 IC50 = 0.5 nM T34296 CY4E9Z 70692916 IC50 > 100000 nM T34296 C0HE2P 70694634 IC50 = 24490 nM T34296 CI8X5B 71449151 IC50 = 4 nM T34296 CMW3O0 71451330 Ki > 200000 nM T34296 CDZ3P2 71453147 Ki = 28 nM T34296 CKW2Q5 71453375 IC50 = 25000 nM T34296 CX3I5C 71458120 IC50 = 17 nM T34296 C3L7SD 71533484 IC50 = 70 nM T34296 CZH5S9 71533485 IC50 = 134 nM T34296 CGM72Q 71540498 IC50 = 11 nM T34296 CXA1I5 71540599 IC50 = 164 nM T34296 C7CV9E 71540600 IC50 = 23 nM T34296 CA4BP6 71540601 IC50 = 648 nM T34296 CMZ3T2 71540715 IC50 = 155 nM T34296 CXY83G 71540716 IC50 = 44 nM T34296 C1ZH2G 71540717 IC50 = 106 nM T34296 CT4UD5 71540831 IC50 = 104 nM T34296 CP7SX8 71540832 IC50 = 225 nM T34296 C9IW7R 71540833 IC50 = 23 nM T34296 CH5J4A 71602247 IC50 = 22 nM T34296 CH53IU 71602248 IC50 = 386 nM T34296 C97EWQ 71602249 IC50 = 220 nM T34296 CNX9B1 71652215 IC50 = 1.5 nM T34296 C7RZN9 71652216 IC50 = 19 nM T34296 C0NTU7 71652382 IC50 = 0.65 nM T34296 CA5XS1 71652383 IC50 = 62 nM T34296 CYS46I 71652677 IC50 = 4500 nM T34296 CX67VE 71654516 IC50 = 5400 nM T34296 C7DMX5 71680709 Ki = 50 nM T34296 CFPM82 71680710 Ki = 27 nM T34296 C9ZOM7 71680866 Ki = 2 nM T34296 CQ68LT 71680868 Ki > 200000 nM T34296 CV3X1T 71682766 Ki = 200 nM T34296 C5EAO8 71682767 Ki = 160 nM T34296 C80EYX 71682913 Ki = 3400 nM T34296 CIBD03 71682914 Ki = 230 nM T34296 C41BYG 71682915 Ki = 15 nM T34296 C93XEI 71682916 Ki = 10 nM T34296 CQ29PJ 71682917 Ki = 100000 nM T34296 CFWN65 71683062 Ki = 28000 nM T34296 C3L4XU 71718301 IC50 = 12.2 nM T34296 C3E2VT 71814508 IC50 = 1.4 nM T34296 CR2L4T 71814509 IC50 = 1.4 nM T34296 CF21LN 71814684 IC50 = 0.69 nM T34296 C4YM2D 71814685 IC50 = 1.8 nM T34296 CZW1P6 71814686 IC50 = 2.7 nM T34296 C5SI6C 71814687 IC50 = 3.6 nM T34296 CDXZ25 71814688 IC50 = 0.88 nM T34296 CIZ7K1 71814857 IC50 = 1.9 nM T34296 C4W9TJ 71814858 IC50 = 2.9 nM T34296 CJH9K3 71814859 IC50 = 4.7 nM T34296 CCMN52 71814860 IC50 = 5.3 nM T34296 CZ9BC5 71814861 IC50 = 1.6 nM T34296 CU28BE 71815035 IC50 = 0.82 nM T34296 C7HN2J 71815036 IC50 = 3.3 nM T34296 CKV2U5 71817094 Ki = 19 nM T34296 CHDS52 71817095 Ki = 10 nM T34296 C5LZH0 71817097 Ki = 1 nM T34296 C50SID 71817098 Ki = 35 nM T34296 CN83DB 71817100 Ki = 6 nM T34296 CDX2F9 72984326 IC50 = 2.17 nM T34296 CUKG79 73292708 IC50 = 9 nM T34296 C5D3CJ 73292709 IC50 = 1 nM T34296 CL69NM 73292710 IC50 = 1 nM T34296 CQ4RO1 73292711 IC50 = 0.05 nM T34296 C7CT2E 73292869 IC50 = 6 nM T34296 CA0LS6 73292870 IC50 = 0.04 nM T34296 CJU3V6 73292871 IC50 = 0.09 nM T34296 C3PGF2 73292872 IC50 = 1 nM T34296 C0O8VM 73292873 IC50 = 0.3 nM T34296 CBR9I5 73293034 IC50 = 0.1 nM T34296 C9FD2C 73293035 IC50 = 3 nM T34296 C7LP5J 73293036 IC50 = 0.07 nM T34296 C9PQG1 73293037 IC50 = 7 nM T34296 C4PF1H 73293038 IC50 = 0.07 nM T34296 CE39WF 73293196 IC50 = 0.1 nM T34296 CU96XE 73293197 IC50 = 1 nM T34296 CGC51Z 73293198 IC50 = 0.7 nM T34296 CC83FW 73293199 IC50 = 0.6 nM T34296 CS6T8M 73293200 IC50 = 0.3 nM T34296 CW5IQ0 73345859 Ki = 3 nM T34296 CS9AY8 73346035 IC50 = 544.6 nM T34296 CSB01W 73346036 IC50 = 47.3 nM T34296 CCV78D 73346037 IC50 = 14 nM T34296 CUDF74 73347568 IC50 = 31.5 nM T34296 CQ7KG2 73347569 IC50 = 8445 nM T34296 C2B4HW 73349096 IC50 = 1080 nM T34296 CK0TR7 73349097 IC50 = 3.8 nM T34296 C57LGA 73349098 IC50 = 5.1 nM T34296 C25SOB 73349251 IC50 = 0.04 nM T34296 CW01EA 73349535 IC50 > 100000 nM T34296 CFV9Q5 73352169 IC50 = 7329 nM T34296 CA2X8C 73352170 IC50 = 17.7 nM T34296 CXT5V1 73352171 IC50 = 1051 nM T34296 C7Z9MF 73352172 IC50 = 1617 nM T34296 C43WKX 73353429 Ki = 1 nM T34296 CK42DO 73353430 Ki = 5 nM T34296 CNW2C8 73353628 IC50 = 71.2 nM T34296 CYV0L6 73353629 IC50 = 13.8 nM T34296 CG6R7T 73353630 IC50 = 6980 nM T34296 C6H5TU 73354941 Ki = 10 nM T34296 C1HLC9 73355128 IC50 = 2.8 nM T34296 CX8HV9 73355129 IC50 = 178 nM T34296 C06BPT 73355130 IC50 = 18.2 nM T34296 C0K9RX 73355131 IC50 = 53.8 nM T34296 CEHB08 73356503 Ki = 323 nM T34296 C4SXT6 73356696 IC50 = 8.3 nM T34296 CA5T7P 73603957 IC50 = 4200 nM T34296 C8VN1R 74221194 IC50 = 1100 nM T34296 CUB7V9 76329513 IC50 = 0.5 nM T34296 C21FEO 76331549 IC50 = 43 nM T34296 CX39OW 76331563 IC50 = 216 nM T34296 C9CY5K 76335167 IC50 = 127 nM T34296 CKD41G 81689861 IC50 = 1000 nM T34296 CUE7G4 86287514 IC50 = 7000 nM T34296 CGQ8F3 86287515 IC50 = 930 nM T34296 CJ37XE 86287516 IC50 = 2500 nM T34296 COV8I9 86291010 IC50 = 1114 nM T34296 CO2FL5 90137145 IC50 = 320 nM T34296 CRT54C 101910871 IC50 = 30000 nM T34296 C1W5NH 118718816 IC50 = 150 nM T34296 C5ZS4E 118722686 IC50 = 720 nM T34296 CIZB24 118722687 IC50 = 3100 nM T34296 C5C0ZX 118722688 IC50 = 4700 nM T34296 CNF86U 121493953 Ki = 0.008 nM T34296 CJFS09 122190237 IC50 = 1800 nM T34296 CF9C4N 127025165 IC50 = 5.37 nM T34296 CH59PY 127025166 IC50 = 93.8 nM T34296 COGJ69 127025217 Ki = 119 nM T34296 CF45SG 127025218 Ki = 110 nM T34296 CD36QJ 127025222 Ki = 4 nM T34296 CO1DJ9 127027301 IC50 = 2.41 nM T34296 CPG8E6 127027350 Ki = 33.6 nM T34296 CXS26T 127027351 Ki = 14.1 nM T34296 CM7B5S 127029507 IC50 = 1030 nM T34296 C6HA8I 127029508 IC50 > 100000 nM T34296 CPM3N2 127029509 IC50 = 73.1 nM T34296 C3B9EY 127029510 IC50 > 100000 nM T34296 CKNI84 127050262 IC50 = 6 nM T34296 CYA92R 130282633 IC50 = 1300 nM T34296 CO3QE2 130282636 IC50 = 1200 nM T34296 CTN42D 132941363 IC50 = 18000 nM T34296 C83FAY 134130294 Ki = 57.5 nM T34296 C9J7UE 134152374 IC50 = 11 nM T34296 CN9D7G 134155756 IC50 = 0.12 nM T34296 C7K4PA 135412054 IC50 = 920 nM T34296 C31VAN 135412231 Ki = 800 nM T34296 C2VKE8 135414653 IC50 = 16500 nM T34296 CHV2U1 135438561 IC50 = 0.0039 nM T34296 CN30DX 135438809 IC50 = 1600 nM T34296 C4FVJ1 135487604 IC50 = 49600 nM T34296 C8R4FB 135546884 Ki = 1526 nM T34296 C6GR3K 135567051 IC50 = 0.2 nM T34296 C1MOD4 135567320 IC50 = 3.4 nM T34296 CZ0NP3 135924162 IC50 = 36 nM T34296 C2R1MP 135982287 IC50 = 1.7 nM T34296 CFX24R 135982332 IC50 = 16 nM T34296 CWP01Y 135982353 IC50 = 9.4 nM T34296 CR2A9D 135982354 IC50 = 29 nM T34296 CQP35S 135982356 IC50 = 65 nM T34296 CAJ75N 135995993 IC50 = 0.03 nM T34296 CASN17 135995994 IC50 = 0.15 nM T34296 C8EWM3 135995995 IC50 = 0.04 nM T34296 CAO12W 135995996 IC50 = 34 nM T34296 C5BO6Y 135995997 IC50 = 0.99 nM T34296 C6VP7Q 135995998 IC50 = 0.16 nM T34296 CG96KF 135995999 IC50 = 2.9 nM T34296 C5QMP6 135996000 IC50 = 9.7 nM T34296 CYOZ82 135996001 IC50 = 4.3 nM T34296 CI8E5D 135996002 IC50 = 1.6 nM T34296 C5PA8K 135996003 IC50 = 0.52 nM T34296 CATJ83 135996004 IC50 = 0.69 nM T34296 CNJ8H9 135996005 IC50 = 0.31 nM T34296 CW6YS4 135996006 IC50 = 0.53 nM T34296 C1Z8HS 135996007 IC50 = 2.2 nM T34296 C4CB9Z 135996008 IC50 = 8.6 nM T34296 CZWJ74 135996009 IC50 = 25 nM T34296 C1P9QA 135996010 IC50 = 5 nM T34296 C3ZNT0 135996011 IC50 > 10000 nM T34296 CH3J7W 135996012 IC50 = 2200 nM T34296 C7FA3X 135996013 IC50 = 6.3 nM T34296 C2EZ0T 135996014 IC50 = 9.8 nM T34296 CM48OV 135996015 IC50 = 23 nM T34296 CS3Y8H 135996016 IC50 = 1.8 nM T34296 CZ3R8J 135996017 IC50 = 110 nM T34296 CVZC21 135996018 IC50 = 27 nM T34296 C29AGZ 136036767 IC50 >= 100000 nM T34296 CMXL16 136036768 IC50 = 25000 nM T34296 C8WP2X 136036769 IC50 = 55880 nM T34296 CO19FB 136036770 IC50 = 89430 nM T34296 CQS0B6 136036777 IC50 = 55880 nM T34296 CU5IK0 136036779 IC50 = 64000 nM T34296 C49YHB 136036783 IC50 >= 100000 nM T34296 CU54MP 136036786 IC50 = 158 nM T34296 C12UID 136036787 IC50 = 32000 nM T34296 CR9Q6H 136054467 IC50 = 1.6 nM T34296 CYH23I 136054468 IC50 = 0.59 nM T34296 CZ8DW1 136054472 IC50 = 0.38 nM T34296 C9H0DL 136054473 IC50 = 1.7 nM T34296 CX7MI0 136054475 IC50 = 0.3 nM T34296 CA5JR6 136054481 IC50 = 0.24 nM T34296 CO2VU9 136054484 IC50 = 0.36 nM T34296 CV47JN 136054485 IC50 = 0.11 nM T34296 CZ48WO 136054487 IC50 = 0.071 nM T34296 CR9CY5 136054490 IC50 = 0.26 nM T34296 C8FGT0 136054495 IC50 = 0.23 nM T34296 CGH39U 136054498 IC50 = 0.19 nM T34296 C2TO7Y 136054508 IC50 = 1.5 nM T34296 CG70BZ 136054516 IC50 = 0.051 nM T34296 CSM57W 136054520 IC50 = 0.052 nM T34296 CXNG40 136118011 Ki > 5025 nM T34296 C1IOH9 136118012 Ki = 4314 nM T34296 CIEW62 136380958 IC50 = 0.17 nM T34296 CHOA14 136814721 IC50 = 26910 nM T34296 CFJ3I6 136814723 IC50 >= 100000 nM T34296 C9HS7J 137287436 IC50 = 0.0032 nM T34296 C4N8VM 137348731 IC50 = 356 nM T34296 CLE8B1 137348732 IC50 = 9.4 nM T34296 C7FQ6W 137348733 IC50 = 2.2 nM T34296 CAZ87R 137631621 IC50 = 35 nM T34296 CQ3GZ0 137632187 Ki = 36 nM T34296 C0I6RH 137632487 IC50 = 1.9 nM T34296 C4KQR9 137635016 Ki = 1.6 nM T34296 C0R5ZT 137635841 IC50 = 32 nM T34296 CU5G8I 137636679 IC50 = 86 nM T34296 C4UMY5 137636781 IC50 = 159 nM T34296 C1RID9 137636861 IC50 = 175 nM T34296 CNM8J4 137638970 IC50 = 5.495 nM T34296 C7Y0FB 137642170 IC50 = 111 nM T34296 CR8H9Z 137644167 IC50 = 4.4 nM T34296 CDOQ29 137644394 IC50 = 36.31 nM T34296 C0Y5JA 137644464 IC50 = 1.6 nM T34296 CB8M6U 137646865 Ki = 1.7 nM T34296 C04KVQ 137647395 IC50 = 14 nM T34296 CK4LE6 137647628 IC50 = 17.9 nM T34296 CHI2E1 137648744 IC50 = 11.75 nM T34296 CXV6J5 137648746 Ki = 0.47 nM T34296 C1U2QR 137651063 IC50 = 25 nM T34296 C9CIY6 137651719 IC50 = 0.3 nM T34296 CZ51XB 137651858 Ki = 24.5 nM T34296 CS80YI 137652598 IC50 = 340 nM T34296 C5Y8RP 137654086 IC50 = 258 nM T34296 CKH37T 137657100 Ki = 190 nM T34296 CZB75K 137657128 IC50 = 16.9 nM T34296 CRD46H 137658344 IC50 = 58 nM T34296 C3ER5O 137658673 IC50 = 128 nM T34296 CEQ8I9 137659945 IC50 = 89 nM T34296 CC3I9B 137660260 Ki = 9.2 nM T34296 CHO70T 137660954 IC50 = 149 nM T34296 C4H0EM 137661370 IC50 = 257 nM T34296 CZ8H6N 137661550 IC50 = 16000 nM T34296 C1IF6L 137661809 IC50 = 20.89 nM T34296 C1Q2BP 145949247 IC50 > 5000 nM T34296 C6TD4M 145949288 IC50 = 2600 nM T34296 CN9RD6 145949408 IC50 = 1200 nM T34296 C5FWA2 145949488 IC50 = 2.5 nM T34296 CZS1N7 145949693 IC50 = 1.9 nM T34296 CYG32L 145950058 IC50 > 5000 nM T34296 CU53BP 145950331 IC50 = 2.5 nM T34296 CY8C4A 145950332 IC50 = 7.8 nM T34296 CAJ25P 145951291 IC50 = 38 nM T34296 C3EF7N 145952515 IC50 = 5.5 nM T34296 CW1GS2 145952760 IC50 = 18.7 nM T34296 CFN1R7 145952843 IC50 = 7.3 nM T34296 CM6T2O 145953417 IC50 = 1300 nM T34296 C6FYK8 145953609 IC50 > 5000 nM T34296 CV80WQ 145954107 IC50 = 9.4 nM T34296 C16VNH 145954604 IC50 = 12.9 nM T34296 CQF50V 145954863 IC50 = 2.4 nM T34296 C8QW9G 145955776 IC50 = 13 nM T34296 CH0ZO5 145955778 IC50 = 14.4 nM T34296 CFDZ62 145955866 IC50 = 2000 nM T34296 CVZ5U7 145955868 IC50 = 6.9 nM T34296 C8TPR1 145956198 IC50 = 43.2 nM T34296 CR8U7Y 145956318 IC50 = 4.4 nM T34296 C4S8LU 145956764 IC50 = 153 nM T34296 CUS0Y9 145957234 IC50 = 9.1 nM T34296 CUO69Q 145957392 IC50 = 88 nM T34296 CX94UK 145957493 IC50 = 289 nM T34296 C6MHN7 145957508 IC50 = 20 nM T34296 C5K7PV 145958060 IC50 = 1.6 nM T34296 CBE02W 145958354 IC50 = 5.1 nM T34296 CQL4O0 145959327 IC50 = 8.5 nM T34296 CUAT97 145960347 IC50 = 18 nM T34296 CZ76WA 145962290 IC50 > 5000 nM T34296 C27MTZ 145962695 IC50 = 148 nM T34296 CRY63E 145963538 IC50 = 6.4 nM T34296 CVCL61 145963739 IC50 = 8.4 nM T34296 C72NJI 145968012 IC50 = 403 nM T34296 CRK13Q 145969600 IC50 = 51 nM T34296 C1FPG2 145972660 IC50 = 6.4 nM T34296 CN73DF 145972870 IC50 = 69 nM T34296 C3F0AD 145973196 IC50 > 2000 nM T34296 CJF73O 145973630 IC50 = 7.1 nM T34296 CX7M9L 145976456 IC50 = 697 nM T34296 CPD1B0 145977213 IC50 = 7.1 nM T34296 C9Z5DX 145978402 IC50 = 274 nM T34296 CZ25LW 155512044 IC50 = 23000 nM T34296 CV10AF 155512426 IC50 = 11 nM T34296 CFHU79 155514943 IC50 = 57 nM T34296 CF64GH 155518335 Ki = 562 nM T34296 CL16UE 155520835 IC50 = 5000 nM T34296 C59YHT 155522902 IC50 = 636 nM T34296 CC5FA9 155529859 IC50 = 4320 nM T34296 CQUA53 155531128 IC50 = 939 nM T34296 C7TP3R 155531151 IC50 > 10000 nM T34296 CJN8X5 155542058 Ki = 1.6 nM T34296 CWEG57 155545190 IC50 = 0.7 nM T34296 C1FP0M 155548067 IC50 = 39 nM T34296 C9AOK6 155550135 IC50 > 10000 nM T34296 C3BA9L 155561798 IC50 = 0.07 nM T34296 CP9YX2 155567218 IC50 = 3400 nM T34296 C8D5VK 155567855 IC50 = 2300 nM T34296 C5U9LI 155569346 IC50 = 280 nM T34296 CLT4Y6 10138589 Ki = 260 nM T34296 C5U3AO 57394286 IC50 = 645 nM T34296 D00KSS 18411961 IC50 = 50 nM T34296 D01OCR 19366856 IC50 = 4 nM T34296 D01UNE 44580457 Ki = 15.7 nM T34296 D02ECA 448942 IC50 = 270 nM T34296 D02EFQ 10549609 IC50 = 16 nM T34296 D02PKO 44294636 IC50 = 500 nM T34296 D03AMR 9849669 Ki = 10 nM T34296 D03FEI 15516781 IC50 = 45 nM T34296 D03SNK 644601 IC50 = 280 nM T34296 D04GOO 10111838 IC50 = 1350 nM T34296 D04UBY 45483018 IC50 = 52000 nM T34296 D04VPH 45376872 IC50 = 4 nM T34296 D05PZV 796420 IC50 = 1700 nM T34296 D05THD 44478925 IC50 = 1400 nM T34296 D07DRT 46175162 Ki = 1.7 nM T34296 D07GEL 10344307 Ki = 0.45 nM T34296 D07MJD 44479701 IC50 = 260 nM T34296 D08ELY 9838786 IC50 = 22 nM T34296 D09GLA 4368 IC50 = 7.943 nM T34296 D09XUQ 19366844 IC50 = 6 nM T34296 D09ZOA 25049753 Ki = 2 nM T34296 D0A0FY 44479457 IC50 = 28000 nM T34296 D0A4TC 446504 Ki = 1.27 nM T34296 D0B3UN 44580458 Ki = 49 nM T34296 D0C1EQ 20348772 IC50 = 95200 nM T34296 D0D7UA 10267279 IC50 = 0.5 nM T34296 D0F4UT 21496278 IC50 = 95900 nM T34296 D0G3YZ 11391583 IC50 = 12000 nM T34296 D0H2PA 9886977 Ki = 0.5 nM T34296 D0H6CK 10160968 Ki > 5025 nM T34296 D0I0WP 649391 IC50 = 13300 nM T34296 D0K0YX 44626352 IC50 = 2450 nM T34296 D0K3RC 44294677 IC50 = 1 nM T34296 D0L6ND 10089677 IC50 = 0.47 ug.mL-1 T34296 D0LB0N 45483008 IC50 > 98000 nM T34296 D0LL8I 9830392 IC50 = 17 nM T34296 D0LM2K 45483015 IC50 = 11300 nM T34296 D0N0FX 19366816 IC50 = 22 nM T34296 D0N6CD 10565532 IC50 = 100 nM T34296 D0NP8A 10370504 IC50 = 73 nM T34296 D0Q4TA 10044321 Ki = 20 nM T34296 D0R5MR 15052873 IC50 = 400 nM T34296 D0S9OL 10155934 IC50 = 2700 nM T34296 D0T1FR 44457233 IC50 > 100000 nM T34296 D0TL3N 45482998 IC50 > 98000 nM T34296 D0V9GS 651854 IC50 = 1300 nM T34296 D0W2UK 6914621 Ki = 1417 nM T34296 D0XE4B 15516780 IC50 = 32 nM T34296 D0XK7G 10445302 Ki = 8 nM T34296 D0Y5IQ 44255320 IC50 = 5000 nM T34296 D0Z7EF 2777 IC50 = 10000 nM T78709 D01AZG 5073 Ki = 21 nM T78709 D01FFA 72301 Ki > 5000 nM T78709 D01ZII 2726 Ki = 673 nM T78709 D03SKR 2803 Ki = 3235.94 nM T78709 D03WEX 9966051 Ki = 9.5 nM T78709 D04JCN 47811 Ki = 1.8 nM T78709 D04JEE 4946 IC50 = 3981.07 nM T78709 D05MBZ 129211 Ki = 0.79 nM T78709 D05XGO 11154555 Ki = 2.6 nM T78709 D05ZIK 4205 Ki > 18 nM T78709 D06FPQ 77992 Ki = 62 nM T78709 D06OSM 91273 Ki = 5.8 nM T78709 D06YFA 31101 Ki = 24 nM T78709 D09IOI 2170 Ki = 221 nM T78709 D0B3UJ 115237 EC50 > 10000 nM T78709 D0CQ0Z 33630 Ki = 356 nM T78709 D0D1AL 3559 IC50 = 1500 nM T78709 D0F2PO 4828 Ki = 22.4 nM T78709 D0G8NN 119570 Ki = 6514 nM T78709 D0H3HM 60795 Ki = 1.7 nM T78709 D0H6QU 6005 Ki = 296 nM T78709 D0H7KF 5002 Ki = 79.43 nM T78709 D0K0KH 656665 Ki = 5.3 nM T78709 D0K0MW 30668 Ki = 125.89 nM T78709 D0K0VO 5639 Ki = 213 nM T78709 D0K8KX 5280343 EC50 > 100000 nM T78709 D0NG7O 60857 Ki = 78.6 nM T78709 D0P0OU 11978813 Ki = 0.12 nM T78709 D0R1JV 60854 Ki = 1.585 nM T78709 D0R6RO 4184 IC50 = 398.11 nM T78709 D0R9EQ 5095 Ki = 1706 nM T78709 D0S9CB 6918248 EC50 = 630.96 nM T78709 D0S9MU 5078 Ki = 140 nM T78709 D0T3KI 4440 Ki = 45 nM T78709 D0T6QX 5736 Ki = 330 nM T78709 D0U2OO 2477 Ki = 3.1 nM T78709 D0UA0I 28693 Ki = 2.3 nM T78709 D0V4QS 135398745 Ki = 610 nM T78709 D0W5HK 216239 Ki = 1181 nM T78709 D0WV3U 4893 Ki > 10 nM T78709 D0X6BV 6918314 EC50 = 0.12 nM T78709 D0X7KB 28864 Ki = 0.4 nM T78709 D0Z1RV 135398737 Ki = 6.38 nM T78709 D0Z6UC 5358 Ki = 230 nM T78709 D01GEB 219050 IC50 = 0.8 nM T78709 D07YVK 9818479 Ki = 73 nM T78709 D09GHO 5311258 Ki = 22 nM T78709 D09IRN 21071390 Ki = 3936 nM T78709 D0F8HS 11741361 EC50 = 389.05 nM T78709 D0HZ2E 5311271 Ki > 10000 nM T78709 D0L3JI 188942 Ki = 180 nM T78709 D0LI1C 44469321 IC50 > 10000 nM T78709 D0N1HW 5311200 Ki = 6620.9 nM T78709 D0P2QO 132787 Ki = 0.7943 nM T78709 D0R9HI 11256720 Ki = 2370 nM T78709 D0T8KA 11151899 Ki = 6.5 nM T78709 D0W5EH 6918388 IC50 < 6 nM T78709 D0X2XF 177336 Ki < 10000 nM T78709 D0Y2GJ 44182694 Ki = 5.05 nM T78709 D0R1PZ 10248159 EC50 = 10 nM T78709 D00OWF 5280953 Ki > 10000 nM T78709 D00KZF 2419 Ki = 0.3715 nM T78709 D01DAW 208951 Ki = 9.3 nM T78709 D01RAE 133079 Ki > 1600 nM T78709 D01VAB 2119 Ki = 21.6 nM T78709 D01WJZ 60820 Ki = 1.7 nM T78709 D02FNU 56971 Ki = 6 nM T78709 D02JMI 9888211 Ki = 2.512 nM T78709 D02VUX 11697676 Ki = 3.7 nM T78709 D02VZP 57347 EC50 = 6.607 nM T78709 D03ITI 183092 Ki = 92 nM T78709 D03QMR 5685 Ki = 2.089 nM T78709 D03TNA 5025739 Ki > 10000 nM T78709 D03ZZH 9887537 Ki = 0.7943 nM T78709 D06DZI 107780 Ki = 70 nM T78709 D07BCO 5684 Ki = 0.1585 nM T78709 D08AWI 11430856 Ki = 5.1 nM T78709 D09WHM 208917 Ki = 1.5 nM T78709 D0B7SP 11292933 Ki = 0.3981 nM T78709 D0EE6L 3038495 Ki = 81 nM T78709 D0G1RT 132059 IC50 = 3.162 nM T78709 D0G5ZL 132792 Ki = 1.9 nM T78709 D0K9JP 9928332 Ki = 2 nM T78709 D0L9SN 4431 Ki = 0.6 nM T78709 D0M7LV 5761 Ki = 1.1 nM T78709 D0O9EM 208928 Ki = 175 nM T78709 D0OS6O 60149 Ki = 33 nM T78709 D0P9FT 148842 Ki = 5.9 nM T78709 D0Q2JS 10436045 Ki = 100 nM T78709 D0R5GS 55191 Ki = 13 nM T78709 D0T1SF 9909448 Ki = 1092 nM T78709 D0Y0RW 66004 IC50 = 5.012 nM T78709 D0YP7L 6604889 Ki < 5 nM T78709 D0Z7AW 9820261 Ki = 180 nM T78709 C5JG6U 2689 IC50 = 46.77 nM T78709 CZUI83 2769 Ki = 794.33 nM T78709 C0H8GR 3191 IC50 = 47 nM T78709 C0OCW6 6240 Ki = 673 nM T78709 C3H5DF 7172 Ki = 63000 nM T78709 C5H9CN 9287 Ki = 3162.28 nM T78709 COD41I 17371 Ki = 256 nM T78709 CVD75F 20810 Ki = 1.3 nM T78709 C9E6DA 21171 Ki > 5000 nM T78709 CFGH18 27620 Ki = 12 nM T78709 C6WDL7 49756 Ki = 200 nM T78709 CPW9B5 65752 Ki > 100000 nM T78709 C06GWQ 72340 EC50 > 100000 nM T78709 CJV28G 90285 IC50 = 2.4 nM T78709 C10XRB 99652 Ki = 32000 nM T78709 CN9GK1 104911 Ki = 0.31 nM T78709 CI24CD 120540 Ki = 43.2 nM T78709 CBS9J2 124433 Ki = 3.58 nM T78709 CI47KZ 127708 Ki = 66 nM T78709 C9WG8X 131559 Ki = 24.8 nM T78709 C4PR2E 132564 IC50 = 8410 nM T78709 CC58NU 132955 Ki = 58 nM T78709 CY0O6P 151779 Ki = 831.76 nM T78709 C4VCM7 156372 Ki = 36000 nM T78709 CI80NA 160436 Ki = 10 nM T78709 CGT8R0 160510 Ki > 1670 nM T78709 C1ND9W 161665 Ki = 149 nM T78709 CK8RD5 168114 Ki = 11710 nM T78709 CJ34CF 168115 Ki = 3740 nM T78709 CLK7P3 169713 IC50 = 3 nM T78709 C3O4NA 179651 Ki > 100000 nM T78709 CZ0D8W 180707 Ki = 2290.87 nM T78709 CA91IX 185559 EC50 > 100000 nM T78709 COPZ85 188006 Ki = 20 nM T78709 C7ASC5 195252 Ki = 19 nM T78709 CQA75X 210165 IC50 = 15 nM T78709 CHLI84 210172 Ki = 1.738 nM T78709 CDA06R 211216 Ki = 181.97 nM T78709 CF72KY 211936 Ki = 1737.8 nM T78709 CJ8XZ3 211938 Ki = 50.12 nM T78709 CVI6X5 213046 Ki = 6.7 nM T78709 C5T7DJ 363353 Ki = 17.5 nM T78709 C2V5FA 398712 Ki = 1 nM T78709 CYV1R3 417052 Ki > 10000 nM T78709 CF7ZS4 417608 Ki = 1.7 nM T78709 C4O6RK 435595 Ki = 830 nM T78709 CFJ3R2 452533 Ki = 90 nM T78709 C0IH9E 688095 Ki = 110 nM T78709 CXQ6U0 735755 IC50 = 7600 nM T78709 C2VLP8 752521 Ki = 660 nM T78709 C5S3MB 785789 Ki > 1000 nM T78709 C1TV2F 1070749 IC50 > 1000 nM T78709 CJ30IQ 1248739 Ki = 3600 nM T78709 C9FI5L 1296368 Ki = 23740 nM T78709 C6VZT7 1984087 Ki = 4900 nM T78709 CGS9R7 2133793 Ki = 13490 nM T78709 CG9N3A 2136365 Ki = 4592 nM T78709 CA2OY6 2737389 Ki = 99 nM T78709 CE50LO 2756712 Ki = 72.1 nM T78709 C1C4LH 2843443 Ki = 26360 nM T78709 C1S8CM 2845719 IC50 > 100 nM T78709 CRA6F5 2853434 Ki = 10330 nM T78709 C3QRD6 2867758 Ki = 31400 nM T78709 CL2G3H 2870750 Ki = 21610 nM T78709 CC74QS 2872937 Ki = 20600 nM T78709 CRF65H 2880253 Ki = 41800 nM T78709 CET7C8 2921525 Ki = 15600 nM T78709 C2DE6R 2927683 Ki = 7100 nM T78709 CF01YE 2928642 Ki = 9100 nM T78709 CY8R6Q 2948971 Ki = 2450 nM T78709 CLXQ01 2950739 Ki = 6100 nM T78709 CO0C7J 2962174 Ki = 284100 nM T78709 CRQ30L 3025767 Ki = 11 nM T78709 CGMD76 3037048 EC50 = 2000 nM T78709 CB5Q2J 3037448 EC50 > 100000 nM T78709 C64CZV 3038494 Ki = 81 nM T78709 CVD51K 3039995 IC50 = 71 nM T78709 C6Z4QI 3050372 Ki = 25 nM T78709 C5NA6S 3069135 Ki = 24 nM T78709 C4X3VL 3073440 Ki = 16 nM T78709 CKB30E 3073449 Ki = 2.099 nM T78709 CAT54M 3074872 Ki = 25 nM T78709 C6SA2G 3132842 Ki = 36800 nM T78709 C82GMT 3246443 Ki = 908 nM T78709 CS8KE2 3649661 Ki = 714 nM T78709 CRUB15 4723431 Ki = 125 nM T78709 C7PX9E 4790508 Ki = 8 nM T78709 CW2C1I 5009938 Ki = 833 nM T78709 C9NKP1 5216959 Ki = 36 nM T78709 CG3Y4K 5221957 IC50 = 2700 nM T78709 C4BKS2 5242341 Ki = 5.3 nM T78709 CY67TC 5281073 Ki = 17 nM T78709 CLNI10 5281408 EC50 = 10300 nM T78709 CH50QK 5281643 Ki > 100000 nM T78709 CZM7D8 5281794 Ki = 18020 nM T78709 CRD82S 5318644 Ki > 100000 nM T78709 C4J3HP 5640104 Ki = 18490 nM T78709 CW34VC 6160690 Ki = 1.3 nM T78709 CCY85T 6442560 Ki = 13050 nM T78709 CFYP06 6442612 Ki = 5840 nM T78709 CWNZ35 6469693 Ki = 2200 nM T78709 CJTQ40 6469918 Ki = 1700 nM T78709 C5K4PX 6603808 Ki = 40.74 nM T78709 CXZ53N 6603866 Ki = 0.1 nM T78709 CP2QM5 6604000 Ki = 151 nM T78709 CR48ZF 6604840 IC50 = 16.9 nM T78709 CC6SM3 6618861 Ki = 354 nM T78709 C0QCK1 6918455 Ki = 398.11 nM T78709 CW0ZE5 6918542 Ki = 702 nM T78709 CC5PQ0 6918601 Ki > 5600 nM T78709 C1WXY3 6918603 Ki = 1000 nM T78709 CD0Z4I 6918648 Ki = 501.19 nM T78709 CX59ZP 6971167 Ki > 100000 nM T78709 C2F3BY 7125890 Ki = 13700 nM T78709 C2PL6S 8019695 IC50 = 9400 nM T78709 C6D0MA 8554729 Ki = 706 nM T78709 CUD06Z 9796627 Ki = 620 nM T78709 C57XYF 9798593 Ki = 0.69 nM T78709 CPG3J9 9798864 Ki = 35.1 nM T78709 CBG80E 9799121 Ki = 90.42 nM T78709 CFC9Y5 9799318 Ki = 512.86 nM T78709 CNE17Q 9799764 Ki = 23.9 nM T78709 CKM1U6 9800010 Ki = 0.2 nM T78709 CJ8SL4 9800133 Ki = 22.4 nM T78709 CSN81W 9801669 Ki = 18.9 nM T78709 CTUX42 9802369 EC50 = 2.138 nM T78709 CCV0M4 9802530 Ki = 40 nM T78709 C2VS1K 9802999 Ki > 1000 nM T78709 CE0DI5 9804612 Ki = 3.981 nM T78709 CNX4F0 9805456 Ki = 1000 nM T78709 CPZ05H 9805881 Ki = 61 nM T78709 CR8ET5 9814387 Ki = 44 nM T78709 CWOS30 9817810 Ki = 140 nM T78709 CX7N8J 9817881 IC50 = 12.59 nM T78709 CHQI10 9818448 Ki = 139 nM T78709 C8S6FJ 9819892 Ki = 1.622 nM T78709 C45QPU 9820163 Ki = 10.9 nM T78709 CS6KM1 9820536 Ki = 170 nM T78709 C1ZM6Q 9821397 IC50 = 2 nM T78709 CD30SC 9821838 Ki = 1.08 nM T78709 CZMK41 9822025 Ki = 5.012 nM T78709 CAX8D6 9822317 EC50 = 1.5 nM T78709 C2U3EZ 9822477 Ki = 69.55 nM T78709 CL2MG5 9822705 Ki = 91.86 nM T78709 CA2D7V 9822812 Ki > 1000 nM T78709 CF0J1A 9822814 Ki = 17.43 nM T78709 C6JN8C 9822942 Ki = 104.1 nM T78709 C5DB6G 9823115 Ki = 29.64 nM T78709 CL38GM 9826580 Ki = 23.4 nM T78709 CPXI10 9826761 Ki = 290 nM T78709 C0AU9L 9826801 Ki = 130 nM T78709 CLU54H 9827354 Ki = 273 nM T78709 CWS18C 9832057 Ki = 17.7 nM T78709 C2MN0P 9837094 Ki > 3521 nM T78709 C6I4QG 9841032 IC50 = 2951.21 nM T78709 C36NME 9842337 Ki = 71.6 nM T78709 C1LOQ2 9842682 Ki = 43.9 nM T78709 C53UPQ 9842861 Ki = 43.65 nM T78709 CXJ7Z3 9844300 Ki = 139.9 nM T78709 C8TE4O 9844321 Ki = 12.07 nM T78709 CFV1I3 9844747 Ki = 2.9 nM T78709 C96YOX 9844821 Ki = 22.2 nM T78709 C4YIM0 9845172 Ki = 248.19 nM T78709 C57TYA 9845202 Ki = 3.5 nM T78709 C5H7TG 9846057 Ki = 549.54 nM T78709 C5MHS3 9847013 Ki = 160 nM T78709 CNB65K 9848303 Ki = 29 nM T78709 CDOG70 9848876 Ki = 236 nM T78709 CYMP40 9851789 IC50 = 1.83 nM T78709 CM13ZV 9856041 EC50 > 10000 nM T78709 C7EZ2L 9859861 Ki > 1000 nM T78709 CZY34F 9860739 Ki = 1.33 nM T78709 C0ZR3E 9861687 IC50 > 100000 nM T78709 CNCK78 9862256 Ki = 170 nM T78709 CC0SQ3 9862968 Ki = 16.8 nM T78709 C8M5XK 9863333 Ki = 899 nM T78709 C6ERH9 9863540 Ki > 3000 nM T78709 CS7EY1 9863750 EC50 = 33.88 nM T78709 CKF2T8 9864325 Ki = 7.5 nM T78709 CTY02P 9865254 Ki = 55 nM T78709 CX3CQ2 9865576 Ki = 75.77 nM T78709 C5WYN4 9865858 Ki = 3.6 nM T78709 C0NV4T 9866094 Ki = 3.981 nM T78709 CHM4D6 9866320 Ki = 3.02 nM T78709 C1SOI8 9867138 Ki = 432.7 nM T78709 CB1F0C 9867475 Ki = 480 nM T78709 C57YPX 9867902 IC50 = 41 nM T78709 C2WB5T 9868306 Ki = 3.12 nM T78709 C8EG1K 9868735 Ki = 1.5 nM T78709 CDFP50 9868793 Ki = 3 nM T78709 C3GMU5 9868889 Ki = 0.2 nM T78709 C7AB8O 9870053 Ki < 3981.07 nM T78709 CHP5L7 9870809 Ki = 12.36 nM T78709 CK76MQ 9872238 Ki = 0.7 nM T78709 CS12TL 9873467 Ki = 18.7 nM T78709 CBF9T3 9879532 Ki = 69 nM T78709 C35LIA 9881324 EC50 = 35 nM T78709 C9NF3D 9881600 Ki = 16 nM T78709 C8L6GE 9882257 Ki > 1000 nM T78709 CY5HZ0 9882594 Ki = 345 nM T78709 C3DB5H 9884781 Ki = 540 nM T78709 CTAC24 9885114 Ki = 792 nM T78709 CW76OG 9885700 Ki = 0.7 nM T78709 COW86S 9886269 Ki = 19.95 nM T78709 CFW03P 9887458 Ki = 134.84 nM T78709 CJW1P5 9888494 Ki = 478.63 nM T78709 C9GB2M 9888555 Ki = 41 nM T78709 C6N8UE 9889681 Ki = 630.96 nM T78709 C1ANB8 9889726 Ki = 122.3 nM T78709 CM52WU 9890119 Ki = 158.49 nM T78709 C2R3PF 9890484 Ki = 214.1 nM T78709 CEG1K5 9891002 Ki = 251.19 nM T78709 C7QMK5 9891617 Ki = 794.33 nM T78709 CEL29O 9891618 Ki = 794.33 nM T78709 C6WY0D 9891901 Ki = 2040 nM T78709 C3J8GU 9892409 Ki = 630.96 nM T78709 CAY78Q 9892644 Ki = 62.22 nM T78709 CAM25C 9894665 Ki = 15 nM T78709 CFM67S 9897637 Ki = 1.66 nM T78709 C9J6KN 9901423 Ki = 4000 nM T78709 CFI97S 9904205 IC50 = 977.24 nM T78709 CUN81Q 9905249 Ki > 10000 nM T78709 CZ32BY 9906183 Ki = 0.54 nM T78709 CYWQ50 9906447 Ki = 432 nM T78709 C25XRA 9906677 Ki > 1000 nM T78709 C7JFZ5 9906978 Ki = 722.3 nM T78709 CWV8K4 9908283 Ki = 52.31 nM T78709 CY2I0L 9908478 Ki = 25 nM T78709 CA4B5Q 9908855 Ki = 5.3 nM T78709 CYZ5N4 9909089 Ki = 0.0631 nM T78709 CWD2G3 9909389 Ki = 0.33 nM T78709 CA0U4Y 9909471 Ki > 1000 nM T78709 CG80QK 9909555 Ki = 76.14 nM T78709 CO7BK6 9909648 Ki = 134 nM T78709 C3BR6W 9910451 Ki = 160 nM T78709 CUX71M 9910468 Ki = 2.9 nM T78709 C4L2CV 9911120 IC50 = 10.72 nM T78709 C9B3EA 9911844 Ki = 316 nM T78709 C78MDV 9913554 Ki = 125.89 nM T78709 CQ3YN1 9927016 IC50 = 12.59 nM T78709 C4UYZ7 9927441 Ki = 520 nM T78709 CY5L0E 9928161 Ki = 804.8 nM T78709 CID4Y2 9928432 Ki = 1.6 nM T78709 CJ6CF2 9928474 Ki = 920 nM T78709 CCX3F8 9929277 Ki = 258.1 nM T78709 CQX4W1 9929572 Ki = 78.3 nM T78709 C7SOT8 9929936 Ki = 275.44 nM T78709 C1C5KY 9931327 Ki = 360 nM T78709 CN3OW2 9932051 Ki = 0.91 nM T78709 CPB27K 9932697 EC50 = 135 nM T78709 C3L5MF 9932835 Ki = 127.84 nM T78709 CN6YW2 9933342 Ki = 0.8 nM T78709 C5V0UE 9933975 Ki = 0.7 nM T78709 C4L1GA 9934033 IC50 = 16.9 nM T78709 CYVZ47 9934284 Ki = 0.3981 nM T78709 CWO45F 9935387 Ki = 199.53 nM T78709 CYH3R7 9947817 Ki = 1000 nM T78709 C63EWV 9950390 Ki = 870 nM T78709 CXUC75 9950482 Ki = 1.6 nM T78709 CP5MQ0 9950538 EC50 = 26 nM T78709 CX6QW8 9952481 Ki = 154.85 nM T78709 C5W6RU 9953959 Ki = 136.45 nM T78709 C4G9VQ 9954092 Ki = 36 nM T78709 CK8NR2 9954121 Ki = 794.33 nM T78709 CU2C3V 9955072 Ki = 0.5 nM T78709 C9QPM4 9955522 Ki = 0.631 nM T78709 CSK1B2 9955819 Ki = 49.5 nM T78709 CHOJ30 9956365 Ki = 128.82 nM T78709 CFR41N 9957068 Ki = 3162.28 nM T78709 CZ9SC7 9957274 Ki = 1.259 nM T78709 CGO64P 9957376 Ki = 3.162 nM T78709 CBK3P7 9958160 Ki = 803.57 nM T78709 C2RU8Q 9966169 Ki = 1100 nM T78709 C9CT0V 9970622 Ki = 81 nM T78709 CR5XJ2 9975609 Ki = 21.6 nM T78709 CCZP34 9976750 IC50 = 5.012 nM T78709 C7JXL1 9976756 Ki = 3.548 nM T78709 C2XG1I 9977716 Ki = 3.162 nM T78709 CFN50J 9978683 Ki > 5000 nM T78709 CPX92V 9979309 Ki = 0.07943 nM T78709 CC6M7Z 9980998 Ki = 27.9 nM T78709 C09GVK 9981322 Ki = 0.75 nM T78709 C2PDI5 9982036 Ki = 2.799 nM T78709 CDG74Q 9983460 Ki = 40.3 nM T78709 CCR0T4 9984109 Ki = 20 nM T78709 CU2EB0 9991334 Ki = 152 nM T78709 CI1OT4 9991554 Ki = 49 nM T78709 CS1DG5 9992098 Ki = 66 nM T78709 CO9EM6 9992630 Ki > 1000 nM T78709 CK54BS 9992778 Ki = 33.9 nM T78709 CF0R6B 9995045 IC50 = 50.12 nM T78709 C3NHU1 9996500 Ki = 2.4 nM T78709 CWQ1K3 9999722 Ki = 10.4 nM T78709 C8A6EZ 10001971 Ki = 0.1259 nM T78709 CVWG72 10003116 Ki = 50.7 nM T78709 CHJ7C0 10003814 Ki = 24 nM T78709 CQL12P 10004545 Ki > 2000 nM T78709 CP54MB 10005122 Ki = 13 nM T78709 C4IG8L 10005161 EC50 = 2.512 nM T78709 CJ4SF5 10005953 Ki = 141 nM T78709 CV4T9U 10008868 Ki = 9.8 nM T78709 CM26VE 10014056 Ki = 54 nM T78709 CO39AR 10014057 Ki = 56 nM T78709 CUX43N 10014136 Ki = 0.1 nM T78709 CG8YK7 10014674 Ki = 1000 nM T78709 CYWH12 10014964 Ki = 5.4 nM T78709 C5MUC9 10015045 Ki = 49 nM T78709 CB32PO 10015338 Ki = 1.5 nM T78709 C3X4BD 10015438 Ki > 1000 nM T78709 C9A2SX 10015574 Ki = 0.12 nM T78709 CS40QN 10015688 Ki = 8.7 nM T78709 CF6OB5 10017429 Ki = 105 nM T78709 CV7R9F 10020040 Ki > 10000 nM T78709 C6XGV2 10020855 Ki = 0.028 nM T78709 CK18LT 10020895 Ki = 56 nM T78709 CQHW51 10023176 Ki = 100 nM T78709 CH6OC0 10024324 Ki = 3.7 nM T78709 CYB6X2 10024776 EC50 = 69.18 nM T78709 CM7W9G 10024936 Ki = 2.512 nM T78709 CR7Y9C 10025854 EC50 = 7.079 nM T78709 CNP9D7 10035788 Ki = 29 nM T78709 CM0Z7A 10036887 Ki > 470 nM T78709 CPXC69 10037436 Ki = 16 nM T78709 C2E1HD 10037437 Ki = 11 nM T78709 C6DT5M 10037522 Ki = 186 nM T78709 CWN9F2 10038106 Ki > 1000 nM T78709 C1IQ5D 10038966 Ki = 9.3 nM T78709 C2C1XS 10042602 Ki = 83.18 nM T78709 CA42DO 10047196 Ki = 9.2 nM T78709 C25WVJ 10047566 IC50 > 1000 nM T78709 C6EDO4 10047814 EC50 = 1.349 nM T78709 C4S0HI 10047915 Ki = 5.2 nM T78709 C2JZL1 10048222 Ki = 8.9 nM T78709 C2UI7F 10048252 Ki > 1000 nM T78709 CF84QJ 10048342 Ki = 0.5012 nM T78709 C8JLO2 10048343 Ki = 0.631 nM T78709 CBF02H 10048892 Ki = 0.247 nM T78709 C3MT0Y 10049499 Ki = 9.9 nM T78709 C4GHO2 10053476 Ki = 125 nM T78709 CFXB93 10059206 Ki = 92 nM T78709 C7CRY4 10059274 Ki = 31 nM T78709 C8KRW5 10059714 Ki = 5.9 nM T78709 C8FT2B 10059787 Ki = 3 nM T78709 C2G9HJ 10060349 Ki > 333 nM T78709 CB96PM 10061032 Ki = 10 nM T78709 CP9A6Q 10061694 IC50 = 63.1 nM T78709 CDA93R 10062435 IC50 = 199.53 nM T78709 C0KWB6 10062885 Ki = 17.3 nM T78709 CJ67EH 10062998 Ki > 1000 nM T78709 CFM51X 10063283 IC50 = 501.19 nM T78709 CUW74G 10064052 Ki = 1420 nM T78709 CR68SH 10064053 Ki = 1.8 nM T78709 C4PCO3 10065083 Ki = 30.5 nM T78709 C0I2RV 10065903 Ki = 3.715 nM T78709 CD0J3I 10067360 EC50 = 2.884 nM T78709 CIC0W2 10068815 Ki = 8.3 nM T78709 C2EG0W 10068933 Ki > 1000 nM T78709 C6HP2C 10069977 Ki = 13.6 nM T78709 C9KWT3 10071738 Ki = 0.3162 nM T78709 CJ50UM 10071897 Ki = 35.97 nM T78709 CT1U0X 10072874 Ki = 426 nM T78709 CV6R2F 10073139 Ki = 0.631 nM T78709 CN9B1F 10074286 Ki = 10.2 nM T78709 CVE2T1 10076176 IC50 = 100 nM T78709 CQ1YA4 10076876 Ki = 6.8 nM T78709 CJ92BN 10082834 Ki = 0.23 nM T78709 CWC26Y 10084026 Ki = 11 nM T78709 CKA5F4 10084076 Ki = 355 nM T78709 CJ16VZ 10084583 Ki = 2500 nM T78709 CD2RM6 10085260 Ki = 960 nM T78709 CQVJ58 10088453 Ki = 79.43 nM T78709 C6BDZ3 10089203 Ki = 460 nM T78709 C6KY5X 10090661 Ki = 29.2 nM T78709 C0IWD7 10091187 Ki = 0.21 nM T78709 C3XY4N 10091300 Ki = 1.023 nM T78709 CW9PL1 10091417 EC50 = 5.248 nM T78709 CR3D5E 10091430 IC50 = 6.31 nM T78709 CJXQ40 10092819 Ki = 17 nM T78709 C7BD6F 10093232 Ki = 39 nM T78709 CR17PA 10093856 Ki = 9.7 nM T78709 C9OXA7 10095692 Ki = 181.97 nM T78709 CLW53J 10097792 Ki = 741.31 nM T78709 CH5WC1 10105311 Ki = 36 nM T78709 C0XO1J 10105844 Ki = 0.2 nM T78709 CB4W8T 10105889 IC50 = 140 nM T78709 CJF84M 10105934 Ki = 1000 nM T78709 C5D2UI 10106412 IC50 = 25.12 nM T78709 C54EYD 10108561 IC50 < 1000 nM T78709 CKU06X 10108730 IC50 = 316.23 nM T78709 CC15UG 10111229 Ki = 83.3 nM T78709 C8CUX9 10112935 Ki = 2.692 nM T78709 CBW28F 10113692 Ki = 58.3 nM T78709 C2ISY6 10114480 Ki = 0.3981 nM T78709 C9PG3D 10115847 Ki = 39.81 nM T78709 CJZX05 10115848 Ki = 1.585 nM T78709 COWN03 10116877 Ki = 1.6 nM T78709 CP1CL5 10127149 Ki = 31.62 nM T78709 CLFA47 10127209 Ki < 10000 nM T78709 CKYQ52 10127424 Ki = 3.981 nM T78709 CRJ8M9 10127673 Ki = 15.85 nM T78709 C4SN0A 10127877 Ki = 2.512 nM T78709 C9J6KH 10128059 Ki = 125.89 nM T78709 CBT24S 10130700 Ki = 400 nM T78709 C8ZJ9G 10131066 Ki = 28 nM T78709 CW0E4F 10137577 Ki = 90 nM T78709 CWMT35 10138727 Ki = 0.7943 nM T78709 C4X9RB 10150658 Ki < 1258.93 nM T78709 CKGC73 10150796 Ki = 158.49 nM T78709 C6FEY0 10151426 Ki = 364 nM T78709 CJI9T7 10151492 Ki = 31.62 nM T78709 C4Q3UL 10154897 Ki > 100 nM T78709 CFL76R 10158326 Ki = 14.3 nM T78709 C3YK0R 10158884 Ki = 5.4 nM T78709 CSPG27 10159927 Ki = 1.585 nM T78709 C9JLX2 10161027 Ki = 19.95 nM T78709 CVA6N0 10161028 Ki = 0.5012 nM T78709 CQEB83 10163855 EC50 > 100000 nM T78709 C5E4SQ 10172853 Ki = 12.59 nM T78709 C3YT8A 10173169 Ki = 398.11 nM T78709 CJRV76 10173263 Ki = 25.12 nM T78709 CMP89S 10173443 Ki = 10 nM T78709 CT0CX5 10174078 Ki = 1.995 nM T78709 CQXI36 10174088 Ki = 2.512 nM T78709 C34ROH 10174199 Ki = 2.512 nM T78709 CG01HR 10178015 Ki = 111.2 nM T78709 CWK76Q 10179327 Ki = 549.54 nM T78709 C4W0PV 10180988 Ki = 6.026 nM T78709 C0NPG1 10180998 Ki = 6.5 nM T78709 COE73R 10183387 Ki = 819.8 nM T78709 CEDP29 10183895 Ki = 0.631 nM T78709 C6NA5G 10194297 Ki = 1000 nM T78709 CI76JU 10194809 Ki = 25.12 nM T78709 CLHY30 10194820 Ki = 251.19 nM T78709 CW1CM3 10195275 Ki = 1 nM T78709 CECA82 10203092 Ki = 1.585 nM T78709 C21MHR 10203336 Ki = 11.3 nM T78709 CE3S6M 10216160 Ki = 398.11 nM T78709 CRW49L 10216744 Ki = 63.1 nM T78709 C80QXD 10216873 Ki = 6.31 nM T78709 C1HF5Y 10222267 Ki = 295 nM T78709 C8LTG3 10223717 Ki = 1.259 nM T78709 C84CPM 10224961 Ki = 2.9 nM T78709 CO57AW 10226822 Ki = 694.2 nM T78709 CF4N1M 10237964 Ki = 1.995 nM T78709 C0Q2ZD 10238160 Ki = 79.43 nM T78709 CIR98N 10238565 Ki = 3.981 nM T78709 CK39BA 10238566 Ki = 2.512 nM T78709 C3L0WD 10238762 Ki = 19.95 nM T78709 CI9KH6 10238763 Ki = 7.943 nM T78709 CAC29B 10243514 IC50 > 1000 nM T78709 CL1K4S 10243702 Ki > 1000 nM T78709 CXD7O8 10244325 Ki = 1.8 nM T78709 CVF1E5 10246054 IC50 > 1000 nM T78709 CSE47M 10247171 IC50 = 5888.44 nM T78709 CG2B7I 10247701 Ki = 125.89 nM T78709 CFCP96 10247720 Ki = 45 nM T78709 C0NT8I 10248163 Ki = 0.31 nM T78709 C4Q2SH 10249573 Ki = 1000 nM T78709 CMA42P 10250834 Ki = 130 nM T78709 CD83JK 10251722 Ki = 390 nM T78709 CUSP67 10252256 IC50 = 17 nM T78709 C4FZ9V 10253106 Ki = 18 nM T78709 C2JDW3 10253939 Ki = 15.9 nM T78709 C4NYW7 10254142 Ki = 22 nM T78709 CX67OE 10254537 Ki = 12.8 nM T78709 CMRA02 10257042 Ki = 7943.28 nM T78709 CZW62U 10262307 Ki = 1000 nM T78709 CG71CB 10263220 Ki > 1000 nM T78709 CXB7U8 10264456 Ki = 721 nM T78709 CI5Z0M 10264555 Ki > 1000 nM T78709 CVT34Y 10264556 Ki > 1000 nM T78709 CC8PX4 10265905 IC50 = 630.96 nM T78709 C10YRB 10266873 Ki = 6.3 nM T78709 CH31DX 10267394 Ki = 2759.7 nM T78709 CR2J1V 10271949 Ki = 83.6 nM T78709 CB95IA 10272536 Ki = 37.15 nM T78709 CC56OL 10272986 Ki = 168.2 nM T78709 C0MVZ1 10273133 Ki = 13 nM T78709 CVC87R 10275633 Ki = 5.012 nM T78709 CL8DY9 10275767 Ki = 563.5 nM T78709 CE9Y8J 10276451 Ki = 198 nM T78709 CQ8N3F 10288132 Ki = 7.943 nM T78709 CWS2U4 10295406 Ki = 4.62 nM T78709 C8XKC0 10310103 Ki = 67 nM T78709 C3G8KJ 10310285 Ki = 5.012 nM T78709 C0WRV9 10310423 Ki = 5.012 nM T78709 CU89JD 10314060 Ki = 405.6 nM T78709 CA3E4W 10316297 Ki = 38.9 nM T78709 CHYJ47 10317514 Ki = 0.79 nM T78709 C5VC9X 10317939 Ki = 13.44 nM T78709 CUT3Y2 10318597 Ki = 24 nM T78709 C0OJ2C 10319235 Ki = 0.5012 nM T78709 CU12DB 10319570 IC50 = 2 nM T78709 CPH30X 10319737 Ki = 0.7943 nM T78709 CCXJ27 10321497 Ki = 42.6 nM T78709 C30CBI 10324625 Ki = 10.2 nM T78709 C3DB1Q 10332122 Ki = 0.5 nM T78709 CMFL49 10332127 Ki = 0.2 nM T78709 CP35VD 10332803 Ki = 19 nM T78709 CFL49K 10333305 IC50 = 125.89 nM T78709 C83GBY 10333405 Ki = 6.1 nM T78709 CE6IP1 10333670 Ki = 178 nM T78709 CRQN68 10333842 Ki = 45 nM T78709 CUY3O1 10340117 Ki = 7.8 nM T78709 CM10QP 10340549 Ki = 607 nM T78709 CXG6B1 10341129 Ki = 0.3981 nM T78709 C4ZI1X 10343002 Ki = 40 nM T78709 C5MH7Y 10343434 Ki = 6.8 nM T78709 C3ZN0F 10344705 Ki = 68.9 nM T78709 CIP38T 10344976 Ki < 1000 nM T78709 CV92JN 10345799 EC50 > 100000 nM T78709 C9IAV3 10346043 Ki > 3162.28 nM T78709 CI17PT 10348924 Ki = 2.2 nM T78709 CH6C8N 10353170 Ki = 11 nM T78709 CS24DU 10353268 IC50 = 287 nM T78709 CXO0J4 10353777 Ki = 4.9 nM T78709 COT48Q 10353846 Ki = 338 nM T78709 CJ6WS4 10354101 Ki = 84.5 nM T78709 C7DQA1 10354437 Ki = 4.7 nM T78709 CUYR47 10355219 Ki = 11 nM T78709 CK7E9M 10355252 Ki = 62.3 nM T78709 C4-DEC 10355779 IC50 = 199.53 nM T78709 CJO3F2 10355844 Ki = 15 nM T78709 CD4H6R 10361512 Ki = 4500 nM T78709 CA4R1B 10362715 Ki = 26.6 nM T78709 COC7M0 10363912 Ki = 0.6026 nM T78709 C72PTA 10364325 EC50 = 229.09 nM T78709 C8GR5I 10364994 Ki = 0.06761 nM T78709 CW41CF 10365352 IC50 = 12 nM T78709 CV0Y5B 10365638 Ki = 39 nM T78709 CR53YS 10365683 Ki = 77.8 nM T78709 C9QBP3 10367560 Ki = 78 nM T78709 CP43QS 10367835 Ki = 10.4 nM T78709 C6ZV2B 10368048 Ki = 7.8 nM T78709 C9LWG3 10369004 IC50 = 38 nM T78709 CD9PZ8 10369020 Ki = 47 nM T78709 CW7MQ0 10376578 Ki = 6.1 nM T78709 CPD3A2 10377136 Ki = 104 nM T78709 C2OWC5 10377224 Ki = 17 nM T78709 CFVW98 10377225 IC50 > 1000 nM T78709 CKMQ51 10377779 Ki = 66 nM T78709 CMJ0B7 10377872 Ki = 1 nM T78709 CIX51R 10378194 Ki = 270 nM T78709 CFT3C8 10378503 Ki = 9.4 nM T78709 CBI62Z 10378937 Ki = 9530 nM T78709 CUV0T8 10379049 IC50 = 316.23 nM T78709 CXQJ16 10379099 IC50 = 316.23 nM T78709 C5LPM8 10379100 IC50 = 316.23 nM T78709 CA7IM5 10379532 Ki = 16.9 nM T78709 CE1XW6 10380005 IC50 = 50.12 nM T78709 CDAC63 10381889 IC50 = 199.53 nM T78709 CMZA83 10383646 Ki > 5000 nM T78709 C69KIB 10385855 Ki = 7.7 nM T78709 CY59KH 10386049 Ki = 0.2884 nM T78709 C0XG9M 10387420 Ki = 0.2512 nM T78709 C8UI9F 10389173 Ki = 1.34 nM T78709 CG1IR6 10394346 Ki = 1.2 nM T78709 C64HBT 10398936 Ki > 470 nM T78709 C3RO4M 10398940 Ki = 174 nM T78709 C0D8HN 10399013 Ki = 4.8 nM T78709 C3LJV4 10400362 Ki = 384 nM T78709 CFEL74 10400539 Ki = 5 nM T78709 C2T0CR 10400849 IC50 = 158.49 nM T78709 CXU73R 10401626 IC50 = 501.19 nM T78709 CVQ9E8 10401691 IC50 = 316.23 nM T78709 CFM13B 10401705 Ki = 8.5 nM T78709 C4L5PQ 10404657 Ki = 499 nM T78709 CHW3Q9 10405775 EC50 = 6.026 nM T78709 CNV6P7 10406539 IC50 = 60 nM T78709 CX72MW 10407711 Ki = 5011.87 nM T78709 CDIZ70 10407753 Ki = 54.59 nM T78709 CU7V2W 10408477 IC50 = 20 nM T78709 CMBW49 10408880 Ki = 15 nM T78709 C8S3XE 10409556 IC50 = 0.1288 nM T78709 CY3O5W 10410577 Ki = 30.55 nM T78709 C01QDW 10411236 EC50 = 1.995 nM T78709 CSH4O3 10411600 Ki = 41.98 nM T78709 C4QJ8U 10412550 Ki = 56 nM T78709 C4TPN1 10413595 Ki = 501.19 nM T78709 CC4QS3 10420841 Ki = 37 nM T78709 C2B0IU 10421236 Ki = 684 nM T78709 C0HM5D 10421583 Ki = 80 nM T78709 CWD56M 10421850 IC50 = 63.1 nM T78709 CYB2Q9 10422079 Ki = 2 nM T78709 C13LGV 10422091 Ki = 2.9 nM T78709 C70IZX 10423337 Ki = 2.9 nM T78709 CR2D4Z 10424079 Ki = 642 nM T78709 CTG0F9 10429067 Ki = 347 nM T78709 CV49RW 10430183 EC50 = 0.78 nM T78709 CR4LS0 10430623 Ki = 573 nM T78709 CD7U5I 10433930 Ki = 3981.07 nM T78709 CK9QE0 10433973 Ki = 30.97 nM T78709 CCP0S9 10434440 Ki = 2.47 nM T78709 CDU91R 10434550 Ki = 257 nM T78709 CPK38Z 10435294 Ki = 46 nM T78709 C4UN0A 10436653 Ki = 69 nM T78709 C8KD1B 10438027 Ki = 130 nM T78709 CSM96F 10443274 Ki = 44 nM T78709 C0Z7FW 10444472 Ki = 145 nM T78709 CBM3X0 10444473 Ki = 69 nM T78709 CMEA74 10445202 Ki = 29 nM T78709 CQ1V2Z 10445845 IC50 = 158.49 nM T78709 CD1FO8 10445902 Ki = 4.1 nM T78709 CBAY90 10445946 Ki = 620 nM T78709 C7VOJ3 10445991 Ki = 15 nM T78709 C9-AUG 10446088 Ki > 1000 nM T78709 C5N8HO 10447116 Ki = 127 nM T78709 CF25ZL 10449555 Ki > 1000 nM T78709 C9WA5Q 10452875 Ki = 1.585 nM T78709 C94TVH 10452995 IC50 = 41686.94 nM T78709 C9YZI1 10453264 EC50 = 7943.28 nM T78709 CFK16Y 10454806 Ki = 0.2512 nM T78709 CYMS64 10454807 Ki = 1.259 nM T78709 C62WSQ 10456474 Ki = 15.1 nM T78709 C10NHR 10457710 Ki = 10 nM T78709 C8V6ZQ 10458087 Ki = 95 nM T78709 CQ4T7G 10458088 Ki = 5.1 nM T78709 CGS4E2 10466294 Ki > 1000 nM T78709 CP17RZ 10466368 Ki = 16 nM T78709 C1YS3M 10466454 Ki = 1000 nM T78709 CK3Q9O 10466960 Ki = 1 nM T78709 CL6FY4 10466962 Ki = 236 nM T78709 C3EH5D 10468253 IC50 = 63.1 nM T78709 COV85C 10472143 Ki = 0.45 nM T78709 C7GEB0 10474042 Ki = 0.08 nM T78709 CUFL05 10474089 EC50 = 2.818 nM T78709 CPI5M7 10476504 Ki = 24 nM T78709 CL63TF 10477223 Ki = 2.512 nM T78709 C8JCZ1 10477386 Ki = 24 nM T78709 CWY2J3 10478217 Ki = 3.981 nM T78709 CEF2O6 10478367 Ki = 641 nM T78709 CE0CF3 10479090 Ki = 100 nM T78709 CI6PN3 10495891 Ki = 19.1 nM T78709 CFQ8U6 10496827 Ki = 19.05 nM T78709 C0QR2H 10496957 IC50 > 100000 nM T78709 C3IY9P 10498554 IC50 = 50118.72 nM T78709 CQ9A2N 10498633 Ki = 1550 nM T78709 C4XWG7 10499348 IC50 = 0.2 nM T78709 C4IXZ5 10500422 Ki = 633 nM T78709 C6TQV3 10501785 IC50 = 0.8 nM T78709 CQE8U0 10502452 IC50 > 100000 nM T78709 CVO4H1 10503335 EC50 = 269.15 nM T78709 C1FV7A 10516340 IC50 = 117.49 nM T78709 CCPO93 10518850 Ki = 18 nM T78709 CTP65K 10519608 IC50 = 2290.87 nM T78709 CWH7R8 10521887 Ki = 90.33 nM T78709 C8WR5O 10522029 IC50 = 0.7 nM T78709 C7M0YQ 10523090 IC50 > 100000 nM T78709 C90TWP 10524876 IC50 = 0.2 nM T78709 CM0BI4 10525991 Ki = 363.08 nM T78709 CNE54K 10526362 IC50 = 389045.14 nM T78709 CDNJ39 10528303 EC50 = 162.18 nM T78709 C8NT2G 10528899 Ki = 5011.87 nM T78709 C5KOM9 10529394 Ki = 1000 nM T78709 C0ZM5P 10531639 Ki = 4 nM T78709 CI67OK 10535587 Ki > 3257 nM T78709 CYKP58 10539093 IC50 = 64565.42 nM T78709 C3N5MZ 10544888 Ki = 2754.23 nM T78709 C48BRW 10546334 Ki = 125.89 nM T78709 CFN8B5 10546440 IC50 = 5370.32 nM T78709 CFC5Z3 10546879 Ki = 109.65 nM T78709 CJ2T5R 10547091 IC50 = 0.3 nM T78709 CTLF72 10547809 IC50 = 102329.3 nM T78709 C1LV7P 10548259 IC50 = 10964.78 nM T78709 C32XGO 10549236 EC50 = 10 nM T78709 C4S7NI 10549573 Ki = 384.59 nM T78709 CJ30TE 10550097 EC50 = 20.42 nM T78709 C3P5VL 10550893 EC50 = 14 nM T78709 COF60K 10550911 EC50 = 8.318 nM T78709 CE59TG 10553922 IC50 > 100000 nM T78709 CYCT15 10562462 Ki = 40.7 nM T78709 CHOZ29 10567450 Ki = 575 nM T78709 C5JY4K 10568666 IC50 > 100000 nM T78709 CW6VX8 10568745 IC50 = 6165.95 nM T78709 CART26 10569395 IC50 = 4570.88 nM T78709 C7N1FY 10569470 IC50 = 257.04 nM T78709 CY37OI 10570263 Ki = 323.59 nM T78709 CQJ29H 10570535 Ki = 12.02 nM T78709 C5YH2I 10571274 Ki = 554 nM T78709 C9GSI8 10571450 IC50 = 12882.5 nM T78709 CN1UG2 10572945 Ki = 501.19 nM T78709 CY05PE 10573164 IC50 = 12589.25 nM T78709 CU63GA 10573576 IC50 = 0.8 nM T78709 CHE80N 10573876 Ki = 398.11 nM T78709 CBZP14 10574764 Ki = 89.13 nM T78709 CZ0IY9 10575934 EC50 = 5.754 nM T78709 CZC23D 10576554 EC50 = 309.03 nM T78709 C61SEA 10576618 IC50 = 17782.79 nM T78709 CM9N5S 10585117 Ki = 120 nM T78709 C69LZJ 10590206 IC50 = 120.23 nM T78709 C0DX7G 10590360 IC50 = 93.33 nM T78709 CCBU34 10590370 Ki = 2300 nM T78709 CV9LP1 10592579 Ki = 794.33 nM T78709 C7EN0K 10593348 Ki = 48.8 nM T78709 C5G1OF 10594234 Ki = 6.7 nM T78709 C9PKO0 10595710 Ki = 416.87 nM T78709 CBT12J 10596337 Ki = 5011.87 nM T78709 CO23YX 10597140 Ki = 1584.89 nM T78709 CW3TN5 10598044 IC50 = 31622.78 nM T78709 C85LBE 10600032 EC50 = 39.81 nM T78709 CO24RV 10600444 Ki = 446.68 nM T78709 CF74VT 10601619 Ki = 13.4 nM T78709 C49WAM 10610641 Ki = 14.4 nM T78709 CVYB63 10613373 Ki = 48 nM T78709 COB4F8 10616442 Ki = 15.85 nM T78709 C76HPC 10616443 Ki = 10 nM T78709 C42HFS 10616657 Ki > 1000 nM T78709 C2G4IR 10617200 Ki = 5.495 nM T78709 CRY9Q0 10617292 IC50 = 2570.4 nM T78709 C8GFT6 10618751 Ki = 27 nM T78709 C7KD2F 10619048 Ki = 18.2 nM T78709 C39FNQ 10619583 IC50 = 89125.09 nM T78709 C86KEZ 10620679 IC50 = 40738.03 nM T78709 CX3A0P 10620719 Ki = 967 nM T78709 CIV3M9 10621014 Ki = 501.19 nM T78709 CQH1X3 10621131 IC50 = 288.4 nM T78709 CD8KX9 10621491 Ki > 3356 nM T78709 CMV72H 10622257 IC50 = 25703.96 nM T78709 CFR74L 10623260 Ki = 19.95 nM T78709 CTA56W 10623356 Ki = 0.791 nM T78709 C6PXH9 10623459 Ki = 549.54 nM T78709 CUH0N7 10623740 Ki = 5011.87 nM T78709 CHO45W 10624365 Ki = 5011.87 nM T78709 CL8K0J 10624420 Ki = 257.04 nM T78709 CEWL87 10624604 Ki = 17.22 nM T78709 C0DZC5 10624695 Ki = 32.81 nM T78709 C01MLV 10637485 IC50 = 117.49 nM T78709 CAPO49 10638372 Ki > 1000 nM T78709 C1MYD5 10640199 Ki = 885 nM T78709 CQ1NJ0 10640504 Ki = 707.95 nM T78709 CER8L0 10640982 Ki = 0.8318 nM T78709 C2FH3S 10643939 Ki > 1000 nM T78709 C1A6ZO 10644514 IC50 = 3 nM T78709 C9XE8T 10645076 IC50 = 3000 nM T78709 CCS31Z 10645335 IC50 = 61659.5 nM T78709 CQD6R2 10645615 IC50 = 660.69 nM T78709 C8HO3D 10646854 Ki = 1584.89 nM T78709 CN5I9Q 10646934 EC50 = 30.9 nM T78709 CU50HJ 10647006 EC50 = 3.467 nM T78709 C6PBY1 10647387 Ki = 1 nM T78709 CPMS86 10647621 EC50 = 14.79 nM T78709 C5KNR9 10647622 EC50 = 2.754 nM T78709 CCA14X 10648046 Ki = 5011.87 nM T78709 CYDV92 10649124 Ki = 14.1 nM T78709 CH3V2L 10661560 Ki = 50.12 nM T78709 CQM6J9 10662302 Ki = 204 nM T78709 C07AKO 10663820 IC50 > 100000 nM T78709 CEVO29 10664203 Ki = 63 nM T78709 C87GYV 10664657 Ki = 199.53 nM T78709 C5W6PY 10665156 Ki = 9.3 nM T78709 CZN9V7 10665419 IC50 = 15488.17 nM T78709 C4PV2W 10666301 IC50 = 6760.83 nM T78709 CB3C9Z 10667071 IC50 = 40738.03 nM T78709 CH37WD 10669519 Ki = 501.19 nM T78709 CNFI24 10670050 EC50 = 6.607 nM T78709 C4D0QG 10671211 IC50 = 2 nM T78709 C4NOI8 10672566 Ki = 42.85 nM T78709 C0U6ZS 10672840 Ki = 114 nM T78709 CBC8N5 10674136 Ki = 5011.87 nM T78709 CC24YZ 10686563 Ki = 794.33 nM T78709 CCZ41N 10687440 Ki = 5011.87 nM T78709 CTS4A1 10687868 IC50 = 33884.42 nM T78709 CBEP65 10688604 Ki = 22.39 nM T78709 CTXW74 10688951 Ki = 33.88 nM T78709 CP45QK 10689339 IC50 = 43651.58 nM T78709 C26GSJ 10689888 Ki = 1000 nM T78709 C4I3YM 10690445 Ki = 50.12 nM T78709 C6YXC1 10691383 IC50 = 11 nM T78709 C5FQ9T 10691904 Ki = 23 nM T78709 C2LU1H 10692095 Ki > 3356 nM T78709 C48BQX 10692498 Ki = 851.14 nM T78709 C8SU4D 10692801 EC50 = 407.38 nM T78709 C0BOG6 10694238 EC50 = 33.11 nM T78709 CZLP81 10694239 EC50 = 3.715 nM T78709 CS35LF 10694660 EC50 = 0.7244 nM T78709 C4LM2C 10695395 EC50 = 8.913 nM T78709 CRB2A1 10695466 EC50 = 28.84 nM T78709 CV7D8G 10696202 Ki = 591.56 nM T78709 C9GR4O 10696705 Ki = 60.26 nM T78709 CM31PB 10696930 Ki = 8.6 nM T78709 CS4JW5 10698929 Ki > 10000 nM T78709 CSB3G8 10704251 Ki = 114 nM T78709 CLZ9F5 10706553 Ki = 31.1 nM T78709 CBE87R 10706626 Ki = 142 nM T78709 C61RTM 10709212 Ki = 371.54 nM T78709 CE7DB9 10710400 Ki = 800 nM T78709 C6M0GA 10711251 Ki = 5011.87 nM T78709 C7C9EY 10712619 Ki = 89.13 nM T78709 C9FAP1 10714457 IC50 = 11481.54 nM T78709 CIBU90 10714509 IC50 = 97723.72 nM T78709 CPW52V 10714712 Ki = 5011.87 nM T78709 CU32PG 10714877 Ki = 19.22 nM T78709 CVS29F 10715484 IC50 = 56234.13 nM T78709 CGO34D 10715991 Ki = 100 nM T78709 CX8K5B 10717072 IC50 = 1 nM T78709 C5NQX4 10717512 IC50 = 72.44 nM T78709 C4TV6C 10718220 EC50 = 12.3 nM T78709 CWV5A9 10718277 IC50 = 0.6 nM T78709 C0USP7 10718592 Ki = 3.4 nM T78709 CVK2T3 10718731 IC50 = 204173.79 nM T78709 CP7CE8 10718870 EC50 = 2.63 nM T78709 CI3V8M 10719425 EC50 = 12.02 nM T78709 CM7N9Q 10719857 IC50 = 7762.47 nM T78709 CUS3R0 10720301 Ki = 9.5 nM T78709 CZH1M4 10735345 Ki = 50.12 nM T78709 CZXG16 10735489 Ki = 199.53 nM T78709 CI0GE8 10737848 IC50 = 407.38 nM T78709 CQV9O7 10738182 Ki = 251.19 nM T78709 C1QJ2F 10738317 Ki > 1430 nM T78709 CY1M6L 10738329 IC50 > 100000 nM T78709 C1Y3KQ 10738599 Ki = 5011.87 nM T78709 C1ZH6B 10739272 IC50 = 1047.13 nM T78709 C7YXW0 10740939 EC50 = 3.631 nM T78709 C6SA9J 10742699 EC50 = 28.18 nM T78709 C96VMI 10743303 EC50 = 22.91 nM T78709 C8YQE1 10743835 Ki = 167.88 nM T78709 CX3FL8 10751317 Ki = 88 nM T78709 CZO1E3 10753377 IC50 = 64.57 nM T78709 C17OFU 10756517 IC50 = 67.61 nM T78709 C62VKE 10758083 Ki = 185 nM T78709 CPQ40M 10759541 IC50 = 3 nM T78709 C3TD1I 10762475 Ki = 173.78 nM T78709 CLJ74B 10764513 EC50 = 5.754 nM T78709 CQB52R 10765698 EC50 = 5.248 nM T78709 CWSA98 10777682 IC50 = 32359.37 nM T78709 C1RG2E 10780842 Ki = 716 nM T78709 C9PB7H 10782548 Ki = 794.33 nM T78709 CZJO64 10782681 Ki = 575 nM T78709 CQ12RP 10783275 Ki = 5011.87 nM T78709 CX70KH 10786335 Ki > 1000 nM T78709 CB7V4A 10787178 Ki = 3630.78 nM T78709 CN98JS 10787547 EC50 = 21.88 nM T78709 C6ISL1 10788207 IC50 = 0.7 nM T78709 C5H1DA 10789000 IC50 = 43 nM T78709 C8Y3OP 10789182 EC50 = 2.951 nM T78709 C2QBM4 10789419 EC50 = 3.02 nM T78709 C1XKJ8 10789756 EC50 = 10.72 nM T78709 COJ20B 10790813 IC50 > 100000 nM T78709 C8Y3TP 10791125 Ki = 117 nM T78709 CNUF06 10791244 Ki = 9.5 nM T78709 CK9O3B 10802304 Ki = 38 nM T78709 C5XKN1 10805222 Ki = 144.54 nM T78709 CZ7J1S 10805599 Ki = 1.84 nM T78709 CWA5J0 10807321 Ki = 139 nM T78709 C83RTC 10807421 Ki = 17.38 nM T78709 C2TDU4 10808641 Ki = 190.55 nM T78709 C8S4PF 10808909 IC50 = 14454.4 nM T78709 CPS68R 10809227 Ki = 10 nM T78709 CL12BA 10809238 IC50 = 40 nM T78709 C4K3SY 10809561 IC50 = 125892.54 nM T78709 CXY1Q0 10809674 Ki = 14.3 nM T78709 C5J4ND 10809876 IC50 = 0.2 nM T78709 CQN8A4 10811876 IC50 = 1348.96 nM T78709 CL0W3S 10812183 EC50 = 13.18 nM T78709 CQX1G6 10813526 Ki = 54.95 nM T78709 CE16DJ 10813865 EC50 = 5.012 nM T78709 C8QGX9 10813901 EC50 = 1.122 nM T78709 CCWH19 10814515 IC50 > 100000 nM T78709 CUI27T 10825325 Ki = 5.05 nM T78709 CT1I7H 10826076 IC50 = 52.48 nM T78709 CHMB58 10827788 Ki = 120.23 nM T78709 CF4KZ1 10827876 Ki = 154.88 nM T78709 CW2LK3 10828231 Ki = 1180 nM T78709 CVA26N 10830318 Ki = 114.82 nM T78709 CJ1D6P 10830587 Ki = 5011.87 nM T78709 CEW6J2 10831102 Ki = 5011.87 nM T78709 C2XE8D 10831313 Ki = 7.586 nM T78709 C5J1HW 10832055 IC50 = 0.7 nM T78709 CN0Z9Y 10833258 IC50 = 83.18 nM T78709 CL0BO9 10834414 IC50 = 63095.73 nM T78709 C8MHZ9 10835110 Ki = 316.23 nM T78709 C53KRN 10835365 EC50 = 20.89 nM T78709 C0MNA5 10836606 Ki = 1.8 nM T78709 C83QOA 10837858 Ki = 2.2 nM T78709 CC8XL5 10838063 Ki = 12.3 nM T78709 C4V3RT 10848041 Ki = 42 nM T78709 CIQS30 10852612 IC50 = 61.66 nM T78709 CBD60Q 10853821 IC50 > 100000 nM T78709 CU6T1Z 10854403 Ki = 5011.87 nM T78709 CM2TG7 10861457 Ki = 1.175 nM T78709 C3HT1X 10861511 Ki = 0.302 nM T78709 CZ31UD 10861880 Ki = 23.44 nM T78709 C9A8KN 10862425 Ki = 19 nM T78709 C8HN1F 10872581 Ki = 38 nM T78709 COHN31 10873456 Ki = 10.23 nM T78709 C70LSM 10880840 Ki = 37.15 nM T78709 CMV36C 10884046 Ki = 14 nM T78709 CRI50E 10885636 IC50 = 1020 nM T78709 C8OYI0 10891048 Ki = 780 nM T78709 C3I1CT 10892762 Ki = 3.77 nM T78709 CN8P5A 10893547 Ki = 67.61 nM T78709 CEUD36 10893672 Ki = 32.1 nM T78709 CB1HY3 10894144 IC50 = 1570 nM T78709 C2L5YE 10895387 Ki = 2.512 nM T78709 C84RHF 10896220 Ki = 3.3 nM T78709 C1RAP3 10904295 Ki = 17 nM T78709 CC74YP 10905186 Ki = 2.138 nM T78709 C0Q7GV 10915350 Ki = 100 nM T78709 CP7QR4 10915592 Ki = 316.23 nM T78709 CP32CE 10916460 Ki = 1000 nM T78709 CBH30I 10916771 Ki = 13.98 nM T78709 CD7QW2 10917316 Ki = 11.24 nM T78709 CL8AG5 10917920 Ki = 24 nM T78709 C2UZ8H 10917953 Ki = 49 nM T78709 C6D7JR 10924369 Ki = 800 nM T78709 CZN8J0 10925382 Ki = 560 nM T78709 C5X1OQ 10926112 Ki = 100 nM T78709 C3S0ND 10926737 Ki = 0.4365 nM T78709 C0N6KJ 10928520 Ki = 322.1 nM T78709 CD2GN7 10937803 Ki = 1.096 nM T78709 CWE3C9 10946905 Ki = 2000 nM T78709 CNB39C 10947658 Ki = 1.1 nM T78709 CE5XK3 10948133 Ki = 0.16 nM T78709 CGA29L 10948660 Ki = 11.48 nM T78709 CW6T1M 10949284 Ki = 0.5248 nM T78709 CTO4Z9 10949698 Ki = 1.48 nM T78709 CY7B6E 10959998 Ki < 1000 nM T78709 CAIJ61 10961351 Ki = 24.12 nM T78709 C86GIP 10971452 Ki = 5.1 nM T78709 CN6BC3 10972931 Ki = 35 nM T78709 C5NRU3 10973768 Ki = 55 nM T78709 CX5M6J 10974101 Ki = 1.6 nM T78709 CF91AG 10980986 Ki = 0.8318 nM T78709 C6IH1J 10990161 Ki = 550 nM T78709 C4QCY1 10992584 Ki = 0.4467 nM T78709 CF93PW 10992707 Ki = 2.188 nM T78709 CC2NG9 10994812 Ki = 1000 nM T78709 CB1ET0 11002686 Ki = 1.514 nM T78709 C7O5UG 11003379 Ki = 64 nM T78709 CJC9K4 11005810 IC50 = 985 nM T78709 CJS79L 11011968 Ki = 1400 nM T78709 CWU25O 11014017 EC50 > 100000 nM T78709 CLPB39 11014063 Ki = 1.288 nM T78709 C2BF0W 11014848 Ki = 13 nM T78709 CN63RC 11016395 Ki = 5.8 nM T78709 CH9GU5 11016418 Ki = 25 nM T78709 C4T8LY 11020695 IC50 = 8650 nM T78709 CSU4T7 11024618 Ki = 200 nM T78709 C14VMA 11025041 Ki = 26.92 nM T78709 C4Y9XK 11033734 Ki = 255 nM T78709 CX73TF 11035452 Ki = 106 nM T78709 CSK8N7 11037469 Ki = 10.47 nM T78709 C7BS5D 11038248 Ki = 40 nM T78709 C0ES3U 11038263 Ki = 51 nM T78709 CZM27Y 11039289 Ki = 7.2 nM T78709 C7ID8S 11043914 Ki = 2 nM T78709 C3G0FH 11046087 Ki = 400 nM T78709 CH9O0P 11046644 Ki = 0.38 nM T78709 CG0J7X 11047115 Ki = 130 nM T78709 C6EBF3 11048769 IC50 = 2080 nM T78709 CC1YO2 11049209 Ki = 33 nM T78709 C5N9GT 11056946 Ki = 350 nM T78709 CFJG64 11059058 IC50 = 4650 nM T78709 C60SDX 11066440 Ki = 520 nM T78709 C0FT4D 11067619 Ki = 72 nM T78709 CWK94J 11068036 Ki = 30 nM T78709 CL6Y9G 11068509 Ki = 98 nM T78709 C4IN6U 11069073 Ki = 4.898 nM T78709 CG41BK 11071079 IC50 = 1140 nM T78709 CUJ4W7 11071135 Ki = 64 nM T78709 C73PTF 11079090 Ki = 0.8511 nM T78709 C4LP9A 11079476 Ki = 17.38 nM T78709 CKVC23 11079928 Ki = 66.07 nM T78709 CUZ38C 11081136 Ki > 1000 nM T78709 CAJ24R 11090903 Ki = 79.43 nM T78709 CZE43W 11091176 Ki = 1.905 nM T78709 CM2BD4 11092112 Ki = 47 nM T78709 CE42CZ 11092142 Ki = 11 nM T78709 CF32NC 11092254 Ki = 76.23 nM T78709 CRU3M5 11110452 Ki = 41 nM T78709 CC3XK5 11110874 Ki = 22.91 nM T78709 C4VRT9 11111280 Ki = 20 nM T78709 C7DE0U 11113605 IC50 = 1110 nM T78709 CTBF50 11120893 Ki = 840 nM T78709 CVE8T3 11121216 Ki = 6.8 nM T78709 CDMI02 11121708 Ki = 42 nM T78709 C61OTF 11122212 Ki = 1.318 nM T78709 C16LCN 11123104 Ki = 3.02 nM T78709 C6G9KQ 11123573 Ki = 45 nM T78709 CJT65Y 11123606 Ki = 134.5 nM T78709 CF68CS 11133288 Ki = 10.72 nM T78709 C7MD3R 11133868 Ki = 10.23 nM T78709 C3ZJK1 11134424 Ki = 11.6 nM T78709 CC0HY8 11135150 Ki = 53.7 nM T78709 CWB0Z2 11138617 Ki = 3000 nM T78709 CJ63BK 11143175 Ki = 0.631 nM T78709 CA7Y5Z 11144555 Ki = 126.72 nM T78709 C73DFT 11145007 Ki = 1.39 nM T78709 CPA0G8 11145333 Ki = 12 nM T78709 C97CQD 11149594 Ki = 12.5 nM T78709 CYS2X0 11154079 Ki > 1000 nM T78709 C0W4OI 11154198 Ki = 0.54 nM T78709 CVS4I2 11154311 Ki > 1000 nM T78709 CCE1Z3 11156949 Ki = 3.4 nM T78709 CL3C0O 11164277 Ki = 190 nM T78709 C1JC7S 11164569 Ki = 12.9 nM T78709 C8CZQ9 11165409 Ki = 5.14 nM T78709 C8ZN3B 11166042 Ki = 272 nM T78709 CY67TG 11175450 Ki = 4.2 nM T78709 C75WKP 11176199 IC50 = 5 nM T78709 CUE3X2 11176459 Ki = 5.37 nM T78709 C0PHV3 11176648 Ki < 1000 nM T78709 C8KSG5 11177435 Ki = 17.6 nM T78709 CK2V3G 11177467 Ki = 86.25 nM T78709 CL49OC 11178730 IC50 < 10 nM T78709 C6CL1Y 11178830 Ki = 1.585 nM T78709 C4V7ZA 11188024 Ki = 67.8 nM T78709 C4PM2A 11188108 Ki = 300 nM T78709 C8SL0F 11189143 Ki = 17.6 nM T78709 C8FHB1 11189412 Ki = 8.22 nM T78709 C8WHY7 11190823 IC50 = 36.4 nM T78709 C0UQ5K 11191047 Ki > 1000 nM T78709 C6O5JF 11196186 Ki = 827 nM T78709 CCX87L 11200086 Ki = 5.25 nM T78709 C9N5QU 11200511 Ki = 170 nM T78709 C4DUK6 11201573 Ki > 10 nM T78709 CDMQ34 11202474 Ki = 196 nM T78709 COI73W 11206997 Ki = 94 nM T78709 CPX23W 11209208 IC50 > 10000 nM T78709 C36BUG 11210745 Ki > 1000 nM T78709 C4J8YG 11211017 Ki = 54 nM T78709 C41FWO 11213062 Ki = 17.7 nM T78709 C7Q4LE 11213399 IC50 < 10 nM T78709 CVXM03 11221557 Ki = 1.3 nM T78709 C6D1MZ 11223004 Ki = 552 nM T78709 CO58DX 11224478 Ki = 160.3 nM T78709 C0H3SU 11232913 Ki = 0.87 nM T78709 CG71SY 11233991 Ki = 40 nM T78709 C27PSA 11234042 Ki = 260 nM T78709 CLYZ97 11234093 Ki = 1.36 nM T78709 CR10CS 11234230 Ki = 1.06 nM T78709 C0UMB4 11234470 Ki > 1000 nM T78709 C6MI9K 11235335 Ki = 398.11 nM T78709 CNV7Y9 11235558 Ki = 26.27 nM T78709 C3NF5Z 11237443 Ki = 69.18 nM T78709 C1YUE4 11237863 Ki = 5.1 nM T78709 CX5TQ9 11245340 Ki = 248 nM T78709 CJCO91 11245732 Ki = 56.3 nM T78709 CNIC31 11245925 Ki = 125.3 nM T78709 CFC3D9 11246169 Ki = 10.7 nM T78709 C6PUQ7 11246478 Ki = 15.8 nM T78709 CCA7F9 11248217 IC50 = 40 nM T78709 CQ0WO7 11248650 Ki = 46.1 nM T78709 C90WSG 11248705 Ki = 2.512 nM T78709 CS5V2R 11249411 IC50 = 0.7 nM T78709 C7QN4J 11250167 Ki > 1000 nM T78709 CAPX71 11259254 Ki = 63.1 nM T78709 CPBA31 11260140 Ki = 19.2 nM T78709 CEWY47 11261072 Ki = 1.2 nM T78709 CIX25J 11268507 Ki = 65.8 nM T78709 CO25MT 11270107 Ki = 39.81 nM T78709 C2JP5V 11270594 Ki = 5.02 nM T78709 CKEJ43 11270912 Ki = 26.15 nM T78709 C8YKS1 11271864 Ki = 160.5 nM T78709 C5LK4Y 11272673 Ki = 1 nM T78709 C27GXZ 11277680 IC50 > 10000 nM T78709 CJ1S4F 11279872 Ki = 525.6 nM T78709 CW13FD 11280199 Ki = 17.1 nM T78709 CFX51L 11280207 Ki = 8.46 nM T78709 C74SDO 11281688 Ki = 234.4 nM T78709 C2CK8D 11291892 EC50 = 150 nM T78709 CHB4E7 11293380 IC50 = 4 nM T78709 CH4EN9 11293572 Ki = 9.3 nM T78709 C4U7GJ 11293591 IC50 > 2000 nM T78709 CR8ZB5 11295359 Ki = 9.2 nM T78709 C57GTA 11299968 IC50 > 10000 nM T78709 C1VNU0 11303180 Ki = 3.84 nM T78709 CE03YG 11303253 Ki = 2.33 nM T78709 CG0A3L 11303781 Ki = 22.4 nM T78709 C5IQV0 11304135 Ki = 11.27 nM T78709 C9BLC7 11304596 Ki = 0.3981 nM T78709 CJS9C0 11304851 IC50 > 3200 nM T78709 CWF6A1 11305391 IC50 < 10 nM T78709 CI79LV 11307899 Ki = 0.0631 nM T78709 CUXZ91 11311148 IC50 > 10000 nM T78709 C2GZD3 11311204 IC50 > 10000 nM T78709 C9E8WN 11311421 Ki = 252 nM T78709 CI5YQ9 11311820 Ki = 108 nM T78709 C2S0GP 11313610 Ki = 2.5 nM T78709 CCJF50 11313754 Ki = 7.7 nM T78709 CO6NX8 11315660 Ki = 19.97 nM T78709 C1CW4J 11316258 Ki > 10000 nM T78709 CP5E6Q 11316467 IC50 = 3 nM T78709 C0ZXF1 11325675 Ki > 1000 nM T78709 CJT02X 11326158 Ki > 1000 nM T78709 CKUG30 11327798 Ki = 330 nM T78709 CP4K5G 11328306 IC50 < 10 nM T78709 CTN62X 11328382 Ki = 2.512 nM T78709 CBO7W4 11329644 IC50 = 5.2 nM T78709 CH5NT3 11330481 Ki = 8.6 nM T78709 CT3V5I 11338314 Ki = 24 nM T78709 C3JBI0 11338418 Ki > 1000 nM T78709 CT3E6Q 11339067 Ki = 58 nM T78709 C3UA0O 11339351 Ki = 4.07 nM T78709 C4DV2B 11339853 IC50 < 10 nM T78709 CP6VZ2 11339973 Ki = 4.8 nM T78709 CG93PV 11348796 Ki = 25.9 nM T78709 CL7O2I 11349674 Ki = 54.2 nM T78709 C1EGH7 11350339 Ki = 1.68 nM T78709 C8V7GR 11350440 Ki = 717 nM T78709 CJT5E1 11350623 Ki = 26 nM T78709 CI2P0H 11350756 Ki = 19.82 nM T78709 CCY23Q 11351639 Ki = 388 nM T78709 CENY72 11360254 Ki > 1000 nM T78709 CGD42N 11361090 Ki = 97 nM T78709 C6OB5A 11361175 Ki = 29.2 nM T78709 C2HVQ5 11362047 IC50 = 1 nM T78709 CX6N8K 11368804 Ki = 350 nM T78709 CTB03C 11372228 Ki = 9.38 nM T78709 CY20HV 11372576 Ki > 1000 nM T78709 C6A9TH 11373342 Ki = 19.4 nM T78709 CV5XE3 11373704 Ki = 3.5 nM T78709 C1B8WJ 11374059 Ki > 1000 nM T78709 CU6CR4 11374124 IC50 < 10 nM T78709 C2N6CR 11374428 Ki = 2.1 nM T78709 CS9D3C 11374767 Ki = 17.8 nM T78709 CWV4P8 11375860 IC50 > 1000 nM T78709 C5X9JD 11381753 EC50 = 1.3 nM T78709 C6HFW9 11382841 EC50 = 0.34 nM T78709 CHQ9V1 11383270 Ki = 1.94 nM T78709 CBV52J 11384146 Ki = 200 nM T78709 CO1I8H 11384634 Ki = 7.5 nM T78709 CJQ71D 11384983 Ki = 1.29 nM T78709 C3IJD5 11385494 Ki = 73.8 nM T78709 C7XOK1 11394095 Ki = 8.5 nM T78709 CZ2GN9 11394353 Ki = 85.4 nM T78709 C6CAV8 11394411 Ki = 9.8 nM T78709 CU35HP 11395651 Ki = 2.4 nM T78709 CJLS45 11395842 Ki > 1000 nM T78709 CF4OX6 11397149 Ki = 3.981 nM T78709 C7GXP9 11397799 Ki = 6.05 nM T78709 C3V7NH 11405584 Ki = 172 nM T78709 C6WM2A 11406043 Ki > 1000 nM T78709 CMI90K 11407131 Ki > 1000 nM T78709 C7CX1Z 11407133 Ki = 445 nM T78709 CCA2X4 11407766 Ki < 10000 nM T78709 CGN10L 11408148 Ki = 58.8 nM T78709 C6GN7W 11416598 Ki = 36.1 nM T78709 CE5C4L 11418868 Ki = 7.3 nM T78709 C7W6OY 11418949 Ki = 399.2 nM T78709 CKL9J7 11419978 Ki = 1 nM T78709 CRH2D8 11428089 Ki = 1.5 nM T78709 CKPF10 11428376 Ki = 56.3 nM T78709 C13FKL 11429464 Ki > 1000 nM T78709 C0MRK1 11430182 Ki = 3.37 nM T78709 C85LYP 11430418 Ki = 0.7008 nM T78709 C7QX9L 11431037 Ki > 1000 nM T78709 C2B9FV 11440556 Ki = 57.2 nM T78709 CI6NJ2 11440679 Ki = 599.02 nM T78709 C9BNX8 11440979 Ki > 1000 nM T78709 CE79WO 11441652 Ki = 12.08 nM T78709 CGYC26 11442723 Ki = 372 nM T78709 CTD73K 11444410 Ki = 1.9 nM T78709 C6GXJ4 11451971 Ki > 1000 nM T78709 C59SDF 11452106 Ki = 10.1 nM T78709 CM6WJ3 11452107 Ki = 3.3 nM T78709 C6SVK9 11452692 Ki = 2.4 nM T78709 CZ6A2S 11453476 Ki > 1000 nM T78709 C5SJ8M 11459998 Ki = 102 nM T78709 CT73UV 11463955 Ki = 15.6 nM T78709 CG4ST6 11464355 Ki = 794.33 nM T78709 CN6F9K 11464531 IC50 < 10 nM T78709 C89FRU 11464777 Ki = 206.96 nM T78709 C74VWD 11464917 Ki = 107 nM T78709 C6OVE5 11474152 Ki = 25.35 nM T78709 CUOB81 11474564 Ki = 2363.1 nM T78709 C7ZYN5 11474777 Ki = 66.3 nM T78709 C6UBN9 11474937 Ki = 1.2 nM T78709 CQL2E8 11475828 Ki > 1000 nM T78709 CCGF98 11476072 Ki = 398.11 nM T78709 COMY40 11476372 IC50 < 10 nM T78709 CZ5SF1 11477432 IC50 = 91.5 nM T78709 C3QOL9 11484260 Ki = 48 nM T78709 C0GI9R 11484778 Ki = 91.4 nM T78709 CK54EC 11485068 Ki = 5.8 nM T78709 C51OVT 11485631 Ki = 259.34 nM T78709 CC7O5G 11485868 Ki = 2.3 nM T78709 C0XJ1E 11485956 Ki = 41.5 nM T78709 CH9QR1 11486099 Ki = 11 nM T78709 CVX8M3 11486499 Ki = 477.8 nM T78709 C8Q1LZ 11486511 Ki = 0.34 nM T78709 C3NF7L 11487449 Ki = 400.91 nM T78709 C8FN2P 11494093 Ki = 3 nM T78709 C9TU8S 11495769 Ki = 28 nM T78709 CASD80 11501253 Ki = 3 nM T78709 C16AXW 11501537 Ki = 36 nM T78709 CN63TR 11504230 Ki = 25 nM T78709 CE62TB 11511267 Ki = 8.9 nM T78709 CRG4D8 11515921 Ki = 9.31 nM T78709 C59SCV 11516033 Ki = 2300 nM T78709 CW68BJ 11518143 IC50 = 1000 nM T78709 C1KL7T 11518341 Ki = 1.3 nM T78709 CD03GT 11524646 Ki = 112 nM T78709 C38QFE 11530118 IC50 > 10000 nM T78709 CI8GN0 11532563 Ki = 30.9 nM T78709 C7DBO0 11537385 Ki = 52 nM T78709 C0MF3O 11539392 Ki = 11.22 nM T78709 C5ZY6N 11545813 Ki = 2332 nM T78709 C9VC7O 11551780 IC50 > 10000 nM T78709 CW17TM 11554167 Ki = 1.1 nM T78709 COC6U3 11554541 Ki = 11.75 nM T78709 C1V5CH 11559090 Ki > 10000 nM T78709 CY5I0U 11559581 Ki = 390 nM T78709 CVP1Q9 11567578 Ki = 8 nM T78709 CD3Z7J 11567928 Ki = 7.9 nM T78709 CNH1K4 11568826 Ki = 4.7 nM T78709 C8NMI4 11575479 Ki = 170 nM T78709 C6JC2T 11580039 IC50 > 10000 nM T78709 C8CU1X 11581237 Ki = 24 nM T78709 C2IE4D 11583392 Ki = 15.49 nM T78709 C6D1MA 11584660 Ki > 630.96 nM T78709 CU45DK 11595209 Ki > 10000 nM T78709 CGX8F6 11596869 Ki > 3020000 nM T78709 C6G7WS 11603119 Ki = 8 nM T78709 CGD62Y 11603486 Ki = 16 nM T78709 CJW9E6 11604548 Ki = 22.39 nM T78709 CCO15W 11609978 Ki = 218 nM T78709 C6JRN0 11619713 Ki = 23.99 nM T78709 CB7M8E 11625642 Ki = 17 nM T78709 C3IHP8 11626704 Ki = 6.607 nM T78709 C9VAI5 11633517 Ki = 18.2 nM T78709 C2YHQ0 11633739 Ki = 0.77 nM T78709 C2OU7Y 11638332 Ki > 10000 nM T78709 C19UMY 11638640 Ki = 85 nM T78709 CH89AK 11639248 Ki = 6 nM T78709 CI8PF4 11642083 Ki = 14.2 nM T78709 CO89VG 11646566 Ki = 385 nM T78709 C9YA0E 11647443 Ki = 6.3 nM T78709 C1HDM5 11653679 Ki = 117.4 nM T78709 CX7FR8 11655728 Ki = 0.1148 nM T78709 CE4FW0 11662306 Ki = 14 nM T78709 C4L7TV 11662592 Ki = 6.5 nM T78709 C9I7KB 11669646 Ki = 17.38 nM T78709 CB4J2V 11675876 Ki = 3.2 nM T78709 C4KUL7 11676638 Ki = 1.9 nM T78709 CMQX39 11676873 Ki = 34 nM T78709 CTK8R9 11678172 Ki = 22 nM T78709 CLV24Z 11682093 Ki = 258 nM T78709 CDV58J 11696813 Ki = 11.9 nM T78709 C1W8NR 11696910 Ki = 360 nM T78709 CKT7L2 11698732 Ki = 1513 nM T78709 CB4H2O 11699469 Ki = 190 nM T78709 CUVL17 11705133 Ki = 23.44 nM T78709 CJL61W 11706497 Ki = 660 nM T78709 C7RAS6 11712250 Ki = 4.786 nM T78709 C7PK3H 11712470 Ki = 20.89 nM T78709 CHK5I2 11712756 Ki = 0.1585 nM T78709 C46QYG 11720062 Ki = 1360 nM T78709 CGO56C 11720302 Ki = 290 nM T78709 CX9VH0 11720815 Ki = 0.3981 nM T78709 C18COQ 11722647 EC50 = 460 nM T78709 C3KU0D 11722772 Ki > 1000 nM T78709 CAF0J1 11725183 IC50 = 15.85 nM T78709 C2ML7T 11725312 IC50 = 5.012 nM T78709 C1N7MO 11725453 Ki = 142 nM T78709 CXYQ40 11725531 Ki = 2200 nM T78709 C3T9XB 11727140 Ki = 2000 nM T78709 C8YF2N 11728240 Ki = 0.5495 nM T78709 CR29GL 11729007 Ki = 0.7413 nM T78709 CP9TE7 11732304 Ki = 1584.89 nM T78709 CR1L6N 11732516 Ki > 1000 nM T78709 CMO0I9 11739679 Ki = 1670 nM T78709 CL7OG6 11739995 EC50 = 9.06 nM T78709 C57IKL 11740526 Ki = 776.25 nM T78709 CG02AK 11740935 Ki = 40 nM T78709 CJ60OP 11742834 Ki = 6.457 nM T78709 CPG15O 11743399 IC50 > 1000 nM T78709 CVP46J 11746122 Ki = 1000 nM T78709 CYV02C 11747350 Ki = 1800 nM T78709 CO8A3W 11750581 Ki = 9.12 nM T78709 C6IQ8O 11751072 Ki = 4.4 nM T78709 CZN37C 11751188 IC50 = 5 nM T78709 C2J7KO 11751611 Ki > 10000 nM T78709 CBNC94 11752512 IC50 < 10 nM T78709 CS68NX 11754336 Ki = 474.24 nM T78709 CG2WS6 11759467 Ki = 40 nM T78709 CR87JI 11773729 IC50 = 8 nM T78709 CJS7P8 11773878 Ki > 1000 nM T78709 CK1C4D 11774585 Ki = 501.19 nM T78709 C4Y6UC 11776081 Ki > 1000 nM T78709 C4KNX5 11777180 IC50 = 398.11 nM T78709 CJ82MT 11777192 Ki = 79 nM T78709 C2T3OV 11777228 IC50 = 316.23 nM T78709 CM9A7S 11777810 IC50 = 31.62 nM T78709 C06HZD 11782656 Ki = 0.86 nM T78709 CW41AO 11784471 Ki = 1.318 nM T78709 CGI2R8 11792032 IC50 = 4897.79 nM T78709 C2TC7F 11792177 Ki = 34.67 nM T78709 CYR2L7 11793287 IC50 = 346.74 nM T78709 CSLO73 11793877 Ki = 338.84 nM T78709 CW41PM 11793943 Ki = 12.88 nM T78709 CJ0R5E 11794066 Ki = 100 nM T78709 CGVY61 11794853 IC50 = 263.03 nM T78709 CC5DX7 11795765 EC50 = 12.59 nM T78709 C8AWF3 11796209 IC50 = 10232.93 nM T78709 CAMY96 11797158 Ki = 2.2 nM T78709 C90MLE 11797241 IC50 = 22908.68 nM T78709 CQRB24 11797416 Ki = 1584.89 nM T78709 C3U7IY 11797644 IC50 = 8.7 nM T78709 C1M3BY 11797762 IC50 = 54954.09 nM T78709 CN2BP0 11797998 Ki = 1.6 nM T78709 CY75KM 11797999 Ki = 4.3 nM T78709 CAI5J9 11798754 Ki = 5011.87 nM T78709 C3D2AU 11798958 Ki = 21.58 nM T78709 CS19AU 11800592 Ki = 4.06 nM T78709 CVM61S 11809531 Ki = 23 nM T78709 CCI4J0 11810279 Ki = 0.7079 nM T78709 CF9T0I 11810310 Ki = 135 nM T78709 C2R3GJ 11812916 Ki = 49 nM T78709 CLO4B9 11820595 Ki = 0.3 nM T78709 C47SPL 11824009 Ki = 660 nM T78709 CVW4B5 11824522 Ki = 31 nM T78709 CT5DQ9 11824789 Ki = 0.7762 nM T78709 C4WPI2 11825110 Ki = 11.75 nM T78709 CJ49VT 11826976 Ki = 13 nM T78709 CE1QZ8 11827039 Ki = 18 nM T78709 C3LKO9 11845453 Ki = 70.4 nM T78709 C0ZR7C 11845636 Ki = 2.14 nM T78709 CDTQ46 11845643 Ki = 266 nM T78709 CJ9D3N 11845645 Ki = 34.9 nM T78709 CO81MR 11845815 Ki = 1.5 nM T78709 CJ4TH0 11845817 Ki = 2.3 nM T78709 CVOC94 11845819 Ki = 2.1 nM T78709 C3L4QY 11845822 Ki = 1.2 nM T78709 CL0OH3 11845824 Ki = 253 nM T78709 CU39AH 11846005 Ki = 33.2 nM T78709 C58BSD 11846181 Ki = 45.2 nM T78709 CNVY54 11846183 Ki = 18.6 nM T78709 C7P8FK 11846185 Ki = 3.2 nM T78709 CX1B6K 11846187 Ki = 0.1 nM T78709 CXLW54 11948707 EC50 = 0.3 nM T78709 C8JQL7 11957735 IC50 > 10000 nM T78709 C8IFT7 11973922 Ki = 5000 nM T78709 C9IH7R 11973925 Ki = 5000 nM T78709 CS7U5H 11973926 Ki = 5000 nM T78709 C7RY5S 11983282 Ki = 37 nM T78709 CSFD67 11995339 Ki = 5000 nM T78709 CPY4W5 12004114 Ki = 276 nM T78709 C4R5OS 12004116 Ki = 1.2 nM T78709 CLN14H 12004141 Ki = 2 nM T78709 CTFA25 12004142 Ki = 0.4 nM T78709 CTAO18 12004197 Ki = 0.54 nM T78709 C16VZX 12004199 Ki = 0.46 nM T78709 C3QXZ6 12004200 Ki = 0.61 nM T78709 CQ4LI3 12004201 Ki = 0.63 nM T78709 CR9S2B 12004223 IC50 = 2.8 nM T78709 CR3F6P 12004224 Ki = 1.8 nM T78709 C8SVB9 12004226 Ki = 0.61 nM T78709 CI7UF0 12004227 Ki = 3.4 nM T78709 C79VMT 12004253 Ki = 2.1 nM T78709 C3AH4Q 12004254 Ki = 3.6 nM T78709 C2AWK9 12004255 Ki = 0.87 nM T78709 CB2O5M 12004280 Ki = 0.47 nM T78709 C1QY2P 12005903 Ki = 12200 nM T78709 CDNK26 12019526 Ki = 53.2 nM T78709 CCLH20 12313091 Ki > 5000 nM T78709 CLC82F 12374770 Ki = 3750 nM T78709 CQ4V3A 12737487 Ki = 180 nM T78709 CFN31J 12840734 Ki = 35.71 nM T78709 C6P7TB 12840735 Ki = 1.09 nM T78709 C3B8LI 12968865 Ki = 2.72 nM T78709 CB8V2N 12968873 Ki = 4.81 nM T78709 C72BFQ 12968875 Ki = 2.93 nM T78709 C8C5KI 12968876 Ki = 4.08 nM T78709 C13WPY 12968877 Ki = 1.34 nM T78709 C2V9FL 13091268 Ki = 27.7 nM T78709 C2VAE5 13091273 Ki = 37.6 nM T78709 CCG14E 13091356 Ki = 123 nM T78709 C1JW2Q 13091358 Ki = 123 nM T78709 CYN95Z 13091359 Ki = 20 nM T78709 C56TQR 13254321 IC50 = 205 nM T78709 CMA46J 13305910 Ki = 2.455 nM T78709 C0N7VC 13318472 Ki = 1 nM T78709 C2WY8Z 13361400 Ki = 24 nM T78709 C8ALK0 13608253 IC50 = 63 nM T78709 C4A9GO 14039979 Ki = 3.87 nM T78709 CV08GM 14378574 Ki > 5000 nM T78709 C4E7NH 14423371 Ki < 1000 nM T78709 C6E5IV 14576389 EC50 > 100000 nM T78709 CRE73S 14933735 Ki = 0.4 nM T78709 C1Y2UX 14944883 Ki = 1000 nM T78709 CTOY96 14944884 Ki = 0.3 nM T78709 CTQ83H 14944886 Ki = 1.4 nM T78709 C48XLF 14944887 Ki > 1000 nM T78709 CGF64U 14944894 Ki = 16 nM T78709 C47FIY 14950445 Ki = 7.6 nM T78709 C74OKN 14950446 Ki = 103 nM T78709 C8RE3J 14950447 Ki = 1.6 nM T78709 CG96YX 14950448 Ki = 1.9 nM T78709 CFS01M 14950449 Ki = 2.7 nM T78709 CY5P1M 14950450 Ki = 5.3 nM T78709 C0VPR6 14950455 Ki = 0.2 nM T78709 CDT8C1 14950456 Ki = 2.8 nM T78709 CJ16HE 15011385 IC50 = 562 nM T78709 C7VAI1 15011772 IC50 > 10000 nM T78709 CO5C4K 15029820 Ki = 3.2 nM T78709 C7X4LQ 15046233 Ki = 30 nM T78709 CBQY50 15057516 EC50 = 1395 nM T78709 CAF40B 15181802 IC50 = 40 nM T78709 CK21HZ 15226949 IC50 = 58.88 nM T78709 C2XUE8 15344574 Ki = 13 nM T78709 CD25UZ 15389642 Ki = 60.3 nM T78709 C8YB3I 15389644 Ki = 5.9 nM T78709 C8US7F 15410404 Ki = 21 nM T78709 CFTI13 15410410 Ki = 16 nM T78709 C4IB3W 15524005 Ki = 425 nM T78709 CPM16F 15548716 Ki = 1 nM T78709 CL6NC0 15548717 Ki = 6 nM T78709 CZ0A1R 15548718 Ki = 1.7 nM T78709 C06WRK 15548720 Ki = 2.2 nM T78709 C39CEG 15548721 Ki = 72 nM T78709 C0LO4Y 15548722 Ki = 2.3 nM T78709 C5Q8YL 15548723 Ki = 2.8 nM T78709 CRI1N9 15548724 Ki = 5.5 nM T78709 CN5XF4 15549328 Ki = 1.1 nM T78709 C1VWH5 15580747 Ki = 5500 nM T78709 CB6RG2 15654388 Ki = 2.9 nM T78709 CSD46O 15665503 Ki = 0.9 nM T78709 C98WHN 15665505 Ki = 1.2 nM T78709 CMK74C 15665506 Ki = 22 nM T78709 CU31EP 15665507 Ki = 17.8 nM T78709 CT6AY8 15665508 Ki = 0.3 nM T78709 CKQ42I 15665509 Ki = 3 nM T78709 C9SF4H 15665510 Ki = 1 nM T78709 CL2J4H 15665516 Ki = 1.6 nM T78709 C0NUO1 15665517 Ki = 0.6 nM T78709 CYC60K 15744955 Ki = 124 nM T78709 C9J5NY 15744956 Ki = 90 nM T78709 CE6J3A 15744957 Ki = 173 nM T78709 CYD2R7 15744959 Ki = 304 nM T78709 CAF6W2 15744960 Ki = 49 nM T78709 CS50LI 15744961 Ki = 933 nM T78709 CY9H7Z 15744962 Ki > 1000 nM T78709 C1T8UG 15744977 Ki = 12 nM T78709 CEZO41 15744985 Ki = 687 nM T78709 C3AXT9 15744989 Ki = 17 nM T78709 C1XKH0 15744991 Ki = 2.4 nM T78709 CD26OR 15744995 Ki = 31 nM T78709 C02THF 15744998 Ki = 3.2 nM T78709 CT2H9J 15745003 Ki = 105 nM T78709 CK8H9R 15745005 Ki = 109 nM T78709 C5S6ZU 15745006 Ki > 1000 nM T78709 CHQ9A5 15745007 Ki = 84 nM T78709 CY96DH 15745008 Ki = 95 nM T78709 C9LGI7 15745009 Ki > 1000 nM T78709 CU9QY8 15745011 Ki = 171 nM T78709 C74YVE 15745012 Ki > 1000 nM T78709 C90BKV 15745014 Ki = 4493 nM T78709 CCM64H 15786488 Ki = 47.86 nM T78709 CTPX97 15803947 Ki = 17 nM T78709 C1JYT9 15937766 Ki = 44 nM T78709 CT12KQ 15980807 Ki = 927 nM T78709 C5HQT6 15980808 Ki = 19 nM T78709 C4JT9L 15980809 EC50 = 54 nM T78709 C76PIS 15980810 Ki = 129 nM T78709 CF4Z2U 15980852 Ki = 966 nM T78709 CZ39MX 15980853 EC50 = 4 nM T78709 C0H7GI 15980854 Ki = 50 nM T78709 CTH2S5 15980895 Ki = 4 nM T78709 CXW37K 15987265 IC50 = 4800 nM T78709 C1LWZ6 16006605 Ki = 91 nM T78709 CK36NS 16006607 Ki = 265 nM T78709 CMZ69G 16007004 Ki = 4 nM T78709 C3M8GJ 16026344 Ki = 2745 nM T78709 C1SR0O 16071847 Ki > 5000 nM T78709 C4CZ6A 16091081 Ki = 0.4 nM T78709 C7UOM4 16092107 Ki = 24 nM T78709 CD3E8L 16093484 Ki = 181 nM T78709 CEW91O 16093485 Ki = 105 nM T78709 CTFM10 16109481 EC50 = 1412.54 nM T78709 C5RY7T 16109482 EC50 = 67.61 nM T78709 CTCG69 16109483 EC50 < 10000 nM T78709 C0HK1Y 16109484 EC50 = 46.77 nM T78709 CC1R5U 16109485 EC50 = 194.98 nM T78709 CO3HR8 16109486 EC50 = 6.457 nM T78709 C2JW4B 16109487 EC50 = 24.55 nM T78709 CS2QA9 16109488 EC50 = 112.2 nM T78709 C4GRY1 16109489 EC50 = 2.63 nM T78709 CQV32M 16109492 EC50 < 10000 nM T78709 CCOR68 16109496 EC50 = 69.18 nM T78709 CLFO01 16109508 EC50 = 1548.82 nM T78709 C4V8US 16109509 EC50 < 10000 nM T78709 CB8SI6 16109510 EC50 = 134.9 nM T78709 CF2A8R 16109511 EC50 = 32.36 nM T78709 CQS4V1 16112801 IC50 > 1000 nM T78709 CZ1WJ4 16117151 Ki = 455 nM T78709 CM32ZX 16117153 Ki = 4347 nM T78709 CXTB90 16117279 Ki = 859 nM T78709 C1F2LS 16118795 Ki > 5000 nM T78709 C69VDS 16118923 Ki = 3011 nM T78709 CZ2IS9 16660294 Ki > 10000 nM T78709 C3JV0P 16718827 IC50 > 1000 nM T78709 C3YN5S 16718917 IC50 = 1142 nM T78709 CJ8Y1H 16718919 IC50 > 10000 nM T78709 CB7G3R 16718920 IC50 > 1000 nM T78709 CM3FT4 16739258 Ki = 29 nM T78709 CT9GP4 16763549 Ki = 19890 nM T78709 CR63LE 17055181 Ki = 195600 nM T78709 C0QX5J 17374371 Ki = 4307 nM T78709 CF25CM 17449900 Ki = 6.8 nM T78709 C0T9ZY 17947861 Ki = 6.31 nM T78709 C42YEX 18133517 Ki = 52610 nM T78709 CI90UP 18133518 Ki = 38290 nM T78709 C7R1IG 18137015 Ki = 1285 nM T78709 C4I1FW 18137017 Ki = 1637 nM T78709 C07EOI 18137020 Ki = 3614 nM T78709 C9PV8A 18180076 IC50 = 57 nM T78709 CHXQ26 18366015 IC50 = 3548.13 nM T78709 C7G3UV 18694165 IC50 = 6.31 nM T78709 CIEM47 18694195 IC50 = 5.012 nM T78709 CZV26X 18694196 IC50 = 0.3981 nM T78709 CYOU05 18922713 EC50 = 0.13 nM T78709 CJH07D 18988813 Ki > 5000 nM T78709 C78NBQ 18988815 Ki > 1000 nM T78709 CVF4R7 18988817 Ki = 4.7 nM T78709 C08HLD 18988835 Ki > 1000 nM T78709 CV08LK 18988846 Ki = 4.4 nM T78709 C96KED 19023504 IC50 = 440 nM T78709 CU8TB3 19041559 Ki = 210 nM T78709 CYJ48A 19066163 Ki = 393 nM T78709 C0BE1M 19066188 Ki = 450 nM T78709 CV5FR6 19066200 Ki = 1000 nM T78709 C4RU6O 19066201 Ki = 700 nM T78709 CN96TB 19066203 Ki = 571 nM T78709 C60SWJ 19066205 Ki = 79 nM T78709 C5MS9T 19066235 Ki = 3000 nM T78709 C6AOE8 19426635 IC50 > 1000 nM T78709 C25YQI 19770958 IC50 > 10000 nM T78709 CQ3JL0 19956256 IC50 = 5754.4 nM T78709 C7T8JC 19958494 Ki > 10000 nM T78709 C6LI5E 19958507 Ki > 10000 nM T78709 CLVT08 19978038 IC50 = 97.72 nM T78709 CF34NC 19978059 IC50 = 9549.93 nM T78709 C7D0PH 20763915 Ki = 4 nM T78709 C10IHJ 21073216 Ki = 52.7 nM T78709 CH8EN1 21073533 Ki = 40.7 nM T78709 C1R0SA 21073563 Ki = 8.5 nM T78709 CBUG29 21073579 Ki = 1.7 nM T78709 C15NJA 21073584 Ki = 13.8 nM T78709 CXMG13 21073587 Ki = 0.95 nM T78709 C57EJD 21073595 Ki = 4.6 nM T78709 CR0D3H 21073606 Ki = 0.84 nM T78709 C60WIT 21073656 Ki = 1.2 nM T78709 C6CQO1 21073658 Ki = 8.4 nM T78709 C1OL3G 21073667 Ki = 3.3 nM T78709 CVT16Y 21073690 Ki = 2 nM T78709 C9GHF5 21073716 Ki = 3 nM T78709 CA24ZJ 21073731 Ki = 1.2 nM T78709 CGP56E 21073788 Ki = 0.78 nM T78709 C6ARE1 21073793 Ki = 1.1 nM T78709 C3KMW4 21073817 Ki = 3.9 nM T78709 CHM64K 21073872 Ki = 11.4 nM T78709 C5O8SN 21268191 Ki = 7.84 nM T78709 CJ63ET 21268208 Ki = 551 nM T78709 CLW5Z0 21268321 Ki = 32 nM T78709 CQ17TR 21460878 IC50 = 31.62 nM T78709 C2JT9X 21460905 IC50 = 1.995 nM T78709 C3T5HF 21509921 Ki = 596 nM T78709 CFN81Q 21527771 Ki = 74 nM T78709 CH59WN 21533446 Ki = 74 nM T78709 C4B0TN 21557475 Ki = 172 nM T78709 CUV0N3 21689040 EC50 = 1.2 nM T78709 CX45FW 21797090 EC50 = 14.79 nM T78709 CT7XG9 21830793 EC50 = 0.1 nM T78709 C9X8PI 22001618 Ki = 476 nM T78709 CYH4J9 22002244 Ki = 3 nM T78709 CBN84K 22065997 Ki = 990.7 nM T78709 C12QOJ 22113436 Ki = 10.6 nM T78709 CD7M8K 22113440 Ki = 6.82 nM T78709 CF8B0D 22113443 Ki = 28.6 nM T78709 CO32YX 22254068 Ki = 478 nM T78709 CNB53V 22321203 Ki = 6530 nM T78709 C2Z0BJ 22326660 Ki = 19.95 nM T78709 CD80PB 22326688 Ki = 0.2512 nM T78709 CJ3P6O 22326704 Ki = 50.12 nM T78709 C6UXL4 22330705 Ki = 19670 nM T78709 CZG9S2 22425072 Ki = 11860 nM T78709 C5SI3U 22464564 Ki = 93.4 nM T78709 CJ6WF3 22464606 Ki = 25.8 nM T78709 CA5BY9 22464614 Ki = 24.2 nM T78709 CQB94R 22464634 Ki = 9.1 nM T78709 CAZ23L 22464649 Ki = 0.7 nM T78709 CJCY98 22464720 Ki = 2.8 nM T78709 CB97XC 22464804 Ki = 11.8 nM T78709 C9MB7K 22464806 Ki = 429 nM T78709 C7DXE6 22464831 Ki = 2.9 nM T78709 C76FEA 22464842 Ki = 2.5 nM T78709 CPD8Q7 22549784 Ki = 12490 nM T78709 CRU1N2 22611622 Ki = 68 nM T78709 C49VCE 22675297 Ki = 0.82 nM T78709 CIC7F6 22675312 Ki = 15.9 nM T78709 CBCK13 22675339 Ki = 1.04 nM T78709 CPU6C8 22675347 Ki = 3.03 nM T78709 C85YGH 22675350 Ki = 0.89 nM T78709 CP41JS 22675387 Ki = 6.46 nM T78709 C5R7JT 22675398 Ki = 23.4 nM T78709 CA02UK 22849991 Ki = 18.7 nM T78709 C5DJR8 22849992 Ki = 2.9 nM T78709 C3RO8S 22864491 Ki = 106 nM T78709 C91NKL 22864495 Ki = 322 nM T78709 C0MZV7 22998900 Ki = 13 nM T78709 CQB20R 23155620 IC50 = 4.2 nM T78709 CZ25WJ 23155621 IC50 = 62.3 nM T78709 CM57CZ 23155625 IC50 = 5.6 nM T78709 CFB0G1 23155644 IC50 = 55.4 nM T78709 C7FQU2 23155650 IC50 < 10 nM T78709 C8Y7LC 23155667 IC50 < 10 nM T78709 C1PX5S 23155676 IC50 = 7.6 nM T78709 CC46FD 23155688 IC50 < 10 nM T78709 CAC0S3 23155689 IC50 = 4.3 nM T78709 C57WEZ 23155758 IC50 < 10 nM T78709 CXHB39 23155770 IC50 < 10 nM T78709 C1OVU4 23155818 IC50 = 1.3 nM T78709 CKQ2Y0 23155825 IC50 = 18 nM T78709 C2NOU7 23155834 IC50 < 1 nM T78709 C75GWQ 23155840 IC50 = 64.6 nM T78709 C1N6SD 23155860 IC50 = 24.4 nM T78709 CTC8Y5 23155869 IC50 = 90.4 nM T78709 CK3PM5 23155885 IC50 > 100 nM T78709 C8XYR2 23155900 IC50 = 13.5 nM T78709 CFG6D5 23155906 IC50 > 100 nM T78709 CQS93U 23155935 IC50 = 6.1 nM T78709 C3P1TG 23155946 IC50 = 66.6 nM T78709 C5LCT7 23155948 IC50 < 1 nM T78709 C6QCL8 23155950 IC50 > 100 nM T78709 C7DQ5C 23155951 IC50 < 1 nM T78709 C7PSB8 23155955 IC50 < 10 nM T78709 CXR3G9 23155963 IC50 = 96 nM T78709 CC1P4X 23155976 IC50 > 100 nM T78709 CJY62P 23155980 IC50 > 100 nM T78709 CH5C7X 23288790 Ki = 2463 nM T78709 C0NI3J 23290944 Ki = 1.21 nM T78709 CL3O0E 23290959 Ki = 33 nM T78709 C57MVP 23369416 Ki = 40 nM T78709 CL46OM 23625239 EC50 = 2041.74 nM T78709 CP47WR 23625381 EC50 = 3630.78 nM T78709 CFE62K 23625383 EC50 = 154.88 nM T78709 C3CJO8 23625384 EC50 = 309.03 nM T78709 C29WCH 23625533 EC50 = 85.11 nM T78709 CW63KP 23625534 EC50 = 42.66 nM T78709 C1N6WM 23625537 EC50 = 10 nM T78709 CMP38W 23625705 EC50 = 89.13 nM T78709 CXD3E6 23625925 Ki = 1513.56 nM T78709 C1YJ7D 23626001 EC50 = 239.88 nM T78709 CCQ4M1 23626164 EC50 = 446.68 nM T78709 CPZV02 23643663 Ki = 167 nM T78709 CX93TK 23643870 Ki = 112 nM T78709 CO4C6M 23653115 Ki = 36.31 nM T78709 CNU2X4 23725134 IC50 > 1000 nM T78709 CQE1N7 23906630 Ki = 23510 nM T78709 CZ0G9H 24069165 EC50 = 10200 nM T78709 CBXC05 24424330 IC50 = 0.6 nM T78709 CQ0KU9 24738459 Ki = 0.0504 nM T78709 C6GBU8 24762221 Ki = 0.7943 nM T78709 C6Z1PX 24768516 Ki = 79.2 nM T78709 C0HO5Q 24768517 Ki = 168 nM T78709 CX7E3K 24768518 Ki = 60 nM T78709 CW3PD4 24768519 Ki = 1196 nM T78709 C9G8ZH 24768520 Ki = 133 nM T78709 C0VPJ8 24768521 Ki = 415 nM T78709 C9UOG8 24768522 Ki = 2500 nM T78709 CSW50R 24768524 Ki = 29.2 nM T78709 CW8N2E 24768525 Ki = 36.4 nM T78709 CCT04Q 24768526 Ki = 194 nM T78709 C0I2HU 24769156 Ki = 99 nM T78709 CD7CV6 24771120 Ki = 8500 nM T78709 CEQY61 24781869 Ki = 1300 nM T78709 C3JSR4 24794436 IC50 > 1000 nM T78709 CJ4RO1 24804774 Ki = 0.631 nM T78709 CK84BF 24804775 EC50 = 0.03162 nM T78709 C1Z3OQ 24804941 Ki = 1.259 nM T78709 C6AE2U 24804942 Ki = 3.981 nM T78709 C1ZYM4 24804943 Ki = 3.981 nM T78709 C9K0CX 24805674 Ki = 97 nM T78709 CZY17F 24805675 Ki = 28 nM T78709 CT10CH 24805872 Ki = 2.6 nM T78709 C9DTE6 24805873 Ki = 0.2 nM T78709 C8L9WD 24805874 Ki = 0.5 nM T78709 C49EDA 24805875 Ki = 0.38 nM T78709 C58RUQ 24805876 Ki = 0.03 nM T78709 C36NFD 24806070 Ki = 22 nM T78709 CA9G8E 24806071 Ki = 0.2 nM T78709 C9QBV5 24806072 Ki = 2.1 nM T78709 C5I1BZ 24806073 Ki = 4.6 nM T78709 CL61TY 24806074 Ki = 0.54 nM T78709 C58AMS 24829343 Ki = 1610 nM T78709 CDC91N 24839550 Ki = 100 nM T78709 CY21RE 24841480 Ki = 1700 nM T78709 C93JWY 24865538 Ki = 25.12 nM T78709 C5F2VL 24865539 Ki = 5.012 nM T78709 CW9N1Z 24865540 Ki = 158.49 nM T78709 C8PXH7 24865541 Ki = 1258.93 nM T78709 CN5VB4 24865542 Ki = 6.31 nM T78709 CPF5E2 24865543 Ki = 25.12 nM T78709 CGDV58 24865724 Ki = 5.012 nM T78709 C3HK0J 24865725 Ki = 2.512 nM T78709 C5TX3M 24865726 Ki = 12.59 nM T78709 C0O6FX 24865727 Ki = 7.943 nM T78709 C98ZIV 24882509 IC50 = 500 nM T78709 C6L7KS 24887518 Ki < 3162.28 nM T78709 CI53SE 24893978 Ki = 38 nM T78709 CAOF91 24894071 IC50 > 10000 nM T78709 C3C0KP 24894134 EC50 > 50000 nM T78709 CX6R0P 24894141 Ki = 1.413 nM T78709 CMN75S 24901425 Ki = 158.49 nM T78709 C9OAG1 24906198 Ki = 28.18 nM T78709 CUY89J 24936155 Ki = 280 nM T78709 C0BP8C 24939244 IC50 > 10000 nM T78709 C8DJG7 24963860 Ki = 4826 nM T78709 C6DO4B 25032525 Ki = 1.1 nM T78709 CR5FX4 25059765 IC50 > 10000 nM T78709 CMVL70 25059766 IC50 > 1000 nM T78709 CED30A 25059770 IC50 > 1000 nM T78709 CJU9Y7 25060021 IC50 > 1000 nM T78709 C36PMH 25060023 IC50 > 1000 nM T78709 CHSB87 25060024 IC50 > 1000 nM T78709 CTI38U 25060119 Ki = 1310 nM T78709 CYJ5G1 25067564 Ki = 4730 nM T78709 C7O8YH 25068794 Ki = 0.149 nM T78709 CZ9SN8 25068797 Ki = 0.102 nM T78709 CL46IP 25068850 Ki = 0.204 nM T78709 CEH7D9 25068903 Ki = 0.243 nM T78709 CB03DL 25068905 Ki = 0.0152 nM T78709 C5ZHN9 25068906 Ki = 0.0447 nM T78709 C0ZJB7 25068907 Ki = 0.0141 nM T78709 C9G7EM 25068908 Ki = 1.54 nM T78709 CZBY61 25068962 Ki = 0.108 nM T78709 CP9G5Z 25068963 Ki = 0.269 nM T78709 CB3F0I 25068964 Ki > 4.04 nM T78709 CCO7B3 25068966 Ki = 1.46 nM T78709 C16ERI 25069015 Ki = 0.179 nM T78709 CZM94A 25069016 Ki = 0.0501 nM T78709 CYZ45N 25069072 Ki = 1.99 nM T78709 CEB96S 25069073 Ki = 1.92 nM T78709 CAI7V1 25069074 Ki = 0.279 nM T78709 C8A3HM 25069121 Ki = 0.74 nM T78709 CG5WX6 25069122 Ki = 6.88 nM T78709 CS8VK1 25069125 Ki = 1.45 nM T78709 CHZB81 25069180 Ki = 1.3 nM T78709 C3W1AX 25069181 Ki = 0.863 nM T78709 CPGZ03 25069239 Ki = 0.671 nM T78709 CT0R3H 25069240 Ki = 0.341 nM T78709 CX5JF4 25069241 Ki < 0.521 nM T78709 C1P4EC 25069242 Ki = 0.88 nM T78709 CCV27I 25069243 Ki = 0.637 nM T78709 C5BR0K 25069297 Ki = 1.77 nM T78709 CU34CX 25069298 Ki = 0.118 nM T78709 C0Z6YL 25069299 Ki = 2.71 nM T78709 C5Z9MA 25069300 Ki = 0.128 nM T78709 C1OGS2 25069301 Ki < 0.205 nM T78709 C53LJG 25069302 Ki < 0.14 nM T78709 CX74UK 25069353 Ki = 3.04 nM T78709 C8F6VC 25069354 Ki = 3.62 nM T78709 C56RCY 25069355 Ki = 4.56 nM T78709 CI7SM5 25069356 Ki = 5.01 nM T78709 C45AHR 25093400 Ki = 13 nM T78709 C0DFW8 25093401 Ki = 37 nM T78709 C67OHQ 25093402 Ki = 275 nM T78709 CXA09P 25107515 Ki = 2.04 nM T78709 CDW7J5 25107516 Ki = 3.7 nM T78709 C81QKN 25107517 Ki = 40 nM T78709 C1QE6A 25107519 Ki = 13 nM T78709 C3VY8O 25107520 Ki = 70 nM T78709 CYE53P 25107578 Ki = 325 nM T78709 CJO1X8 25107579 Ki = 94 nM T78709 C59IVO 25107580 Ki = 53 nM T78709 CMPG74 25107581 Ki = 10.3 nM T78709 CNW7A8 25107582 Ki = 57 nM T78709 CU71RN 25107583 Ki = 29 nM T78709 C8ZM2J 25107647 Ki = 124 nM T78709 CJF71U 25107648 Ki = 95 nM T78709 C6M9LD 25107649 Ki = 12 nM T78709 CEM90Y 25107650 Ki = 139 nM T78709 C2JW3O 25107651 Ki = 8.2 nM T78709 C7M1XT 25107652 Ki = 19 nM T78709 C4ASH8 25107717 Ki = 43 nM T78709 CQ71NR 25107718 Ki = 106 nM T78709 C3NGR5 25108474 Ki = 1.07 nM T78709 C8GW4P 25108475 Ki = 22 nM T78709 C2FY7C 25128757 Ki = 1720 nM T78709 C5NW4M 25129807 Ki > 10000 nM T78709 CAV81B 25130157 Ki = 1780 nM T78709 CF7P2A 25130875 Ki = 38.9 nM T78709 C7P1QS 25130876 Ki = 3.467 nM T78709 C6G5BO 25130877 Ki = 257.04 nM T78709 CL8GD3 25130878 Ki = 53.7 nM T78709 CT78MG 25130879 Ki = 4.169 nM T78709 C7WXA2 25131192 Ki > 1000 nM T78709 C3UVA0 25131193 Ki = 1.413 nM T78709 C0GM3L 25131196 Ki = 147.91 nM T78709 CCWO92 25131197 Ki = 7.586 nM T78709 CFUT35 25131198 Ki = 0.5888 nM T78709 C9P1ZV 25131523 Ki = 229.09 nM T78709 C1Y3TS 25131871 Ki = 416.87 nM T78709 C8CM1N 25131874 Ki = 37.15 nM T78709 CFJ6Y9 25131876 Ki = 0.6607 nM T78709 CNQX42 25132217 Ki = 25.7 nM T78709 C7WE4Y 25132564 Ki = 234.42 nM T78709 C6K1TB 25132565 Ki = 52.48 nM T78709 CJ19KC 25132566 Ki = 6.026 nM T78709 C67QCG 25132869 Ki > 10000 nM T78709 C0J3RD 25138742 Ki = 10.9 nM T78709 C8SPL6 25138902 Ki = 12.6 nM T78709 CSM12R 25138907 Ki = 0.81 nM T78709 CN13MI 25138912 Ki = 3.98 nM T78709 C3LHY5 25138913 Ki = 3.22 nM T78709 CTYC19 25139055 Ki = 6.21 nM T78709 C9JR6E 25139058 Ki = 1.75 nM T78709 C3VNW8 25139062 Ki = 14 nM T78709 C1QHJ5 25139063 Ki = 10.6 nM T78709 CAY54E 25139064 Ki = 5.44 nM T78709 CB8E6J 25139065 Ki = 19.25 nM T78709 C2L3OB 25139066 Ki = 10.78 nM T78709 C5PO7X 25139217 Ki = 1.32 nM T78709 C0A5NK 25139366 Ki = 2.64 nM T78709 C9RO2S 25139374 Ki = 17.35 nM T78709 CS14YK 25139517 Ki = 6.54 nM T78709 C5JWI0 25139643 Ki = 1.19 nM T78709 C6I9FN 25139645 Ki = 26.1 nM T78709 CJ63XC 25139652 Ki = 3.25 nM T78709 C6OCL8 25139785 Ki = 16.6 nM T78709 CA3E2B 25139914 Ki = 9.64 nM T78709 CD69BU 25140055 Ki = 12.83 nM T78709 CP57TN 25140057 Ki = 39.95 nM T78709 CG05CH 25140362 Ki = 1.88 nM T78709 CQO5P0 25140648 Ki = 5.35 nM T78709 CEF59R 25141218 Ki = 6.2 nM T78709 CL84YJ 25141534 Ki = 100 nM T78709 C4FXR9 25141535 Ki = 132 nM T78709 CW2PL7 25155850 Ki = 1130000 nM T78709 C4UXF6 25155851 Ki > 5000000 nM T78709 C65LWZ 25156129 Ki = 2874000 nM T78709 CS3Q4N 25156130 Ki = 1241000 nM T78709 CZ04VO 25156131 Ki = 756000 nM T78709 C6MXE3 25156132 Ki > 5000000 nM T78709 CU5C7V 25156133 Ki = 800000 nM T78709 C65FNY 25156411 Ki > 5000000 nM T78709 CKIH98 25156412 Ki = 656000 nM T78709 C35NHX 25156413 Ki = 558000 nM T78709 C94OIG 25156414 Ki > 5000000 nM T78709 C1IEF6 25156415 Ki > 5000000 nM T78709 CL1B2G 25156416 Ki = 1124000 nM T78709 CUX0F4 25156684 Ki = 1331000 nM T78709 CB4A2S 25156685 Ki > 5000000 nM T78709 CJO48V 25156686 Ki > 5000000 nM T78709 CF27EQ 25156688 Ki = 686000 nM T78709 C8U6PV 25156966 Ki > 5000000 nM T78709 C05TOB 25157253 Ki > 5000000 nM T78709 CYM3H9 25157257 Ki = 331000 nM T78709 CS0E3J 25157260 Ki > 5000000 nM T78709 CQI4S2 25157543 Ki > 5000000 nM T78709 C6Y4AJ 25157546 Ki = 1310000 nM T78709 CKP10W 25157549 Ki > 5000000 nM T78709 C9B0UR 25157845 Ki > 5000000 nM T78709 CX2CP8 25157848 Ki > 5000000 nM T78709 C1XP3Q 25157850 Ki > 5000000 nM T78709 C5J4ES 25158433 Ki = 1308000 nM T78709 COK46A 25158434 Ki = 1409000 nM T78709 CQRL83 25158435 Ki = 1092000 nM T78709 C26IMW 25158436 Ki = 783000 nM T78709 CNO83H 25181488 Ki = 0.6026 nM T78709 CEYF08 25181489 Ki = 0.5888 nM T78709 CI95EF 25192947 Ki > 10000 nM T78709 CDQ70A 25208878 IC50 > 1000 nM T78709 CJ1Z9H 25216680 Ki = 10100 nM T78709 C1T3LR 25218143 Ki = 8720 nM T78709 CPI03N 25218397 Ki = 8670 nM T78709 CL1R3Q 25218401 Ki = 12200 nM T78709 CW07GN 25256855 Ki = 454 nM T78709 CM2T9Y 25263297 Ki = 6400 nM T78709 CFJM71 25263302 Ki = 5600 nM T78709 C15QMB 25263320 IC50 > 1000 nM T78709 CYS8B2 25265257 EC50 = 18 nM T78709 C4MRQ0 27842480 Ki = 2108 nM T78709 CWT9F7 28918670 Ki = 562.34 nM T78709 CHJ35A 32354149 Ki = 2108 nM T78709 C9QGK3 34257212 Ki = 18 nM T78709 CDV36I 37219401 Ki = 1764 nM T78709 CA58DL 41305446 Ki = 9389 nM T78709 CN2CY7 42266246 Ki = 24.7 nM T78709 CI4Q3O 42266677 Ki = 54.3 nM T78709 CDP76A 42266865 Ki = 2.32 nM T78709 CO3LQ2 42267076 Ki = 50.7 nM T78709 CP54VF 42267840 Ki = 24.4 nM T78709 CWOL80 42273326 Ki = 17.8 nM T78709 CG56DF 42388639 IC50 = 4.6 nM T78709 CH5QX6 42389467 IC50 = 39 nM T78709 C32NKC 42605991 EC50 = 30 nM T78709 CX8L2W 42605992 EC50 = 46 nM T78709 CSY8H7 42605993 EC50 = 20 nM T78709 C0XMS9 42605994 EC50 = 17 nM T78709 CHRM07 42606101 EC50 = 30 nM T78709 C7FMV8 42606103 EC50 = 35 nM T78709 C2J3OV 42606104 EC50 = 20 nM T78709 CL7Q0T 42606105 EC50 = 42 nM T78709 CJ7P0D 42606106 EC50 = 54 nM T78709 CR7S3Z 42606222 EC50 = 12 nM T78709 CDEK82 42606334 EC50 = 99 nM T78709 CW30MB 42606335 EC50 = 50 nM T78709 CY10AG 42606336 EC50 = 62 nM T78709 C6VP2A 42606337 EC50 = 240 nM T78709 CD61JW 42606339 EC50 = 10 nM T78709 CJA90T 42606340 EC50 = 130 nM T78709 C83KBX 42606455 EC50 = 39 nM T78709 CB06ST 42606456 EC50 = 59 nM T78709 CEKO32 42606457 EC50 = 86 nM T78709 C3A6UH 42606458 EC50 = 63 nM T78709 C84YQR 42606459 EC50 = 15 nM T78709 CCZG96 42606461 EC50 = 240 nM T78709 C47AMD 42606572 EC50 = 34 nM T78709 C0TN5O 42606573 EC50 = 16 nM T78709 C1ZD2B 42606577 EC50 = 93 nM T78709 CO59TU 42606688 EC50 = 310 nM T78709 CA0B9F 42625181 Ki = 18.1 nM T78709 C3L0TN 42625183 Ki = 39 nM T78709 CW0OU4 42625185 Ki = 26 nM T78709 CHY12B 42625186 Ki > 1000 nM T78709 CP5X3K 42625188 Ki = 181 nM T78709 C8QSX3 42625267 Ki > 1000 nM T78709 CTM69J 42625269 Ki > 1000 nM T78709 CYM0J6 42625295 Ki = 58.3 nM T78709 CPDG98 42625353 Ki > 1000 nM T78709 CK3QD2 42625354 Ki = 360 nM T78709 CJ64FG 42625356 Ki = 11.5 nM T78709 C27KEF 42625359 Ki > 1000 nM T78709 CN81SE 42625440 Ki = 219 nM T78709 CF7DM0 42625445 Ki = 22 nM T78709 CJI51X 42625446 Ki = 16 nM T78709 CD9RN1 42626103 Ki = 193 nM T78709 CLH7Y0 42626289 Ki > 1000 nM T78709 C75QPL 42626291 Ki > 1000 nM T78709 C5VTZ6 42626293 Ki = 124 nM T78709 C70SWL 42626361 Ki > 1000 nM T78709 CV2X5B 42635027 IC50 = 44 nM T78709 CS9Q3H 42635204 IC50 = 29 nM T78709 CQ2M5S 42635387 IC50 = 215 nM T78709 CR3KM7 42635388 IC50 = 39 nM T78709 CJ3NP5 42636941 IC50 = 5011.87 nM T78709 C8A2VG 43066988 Ki = 30 nM T78709 C0AI7N 43229249 Ki = 707.95 nM T78709 CW2DP3 44123711 Ki = 5.129 nM T78709 C1YM3D 44131466 Ki = 24 nM T78709 CMTB93 44131470 Ki = 29 nM T78709 CYE20L 44131666 Ki = 3.7 nM T78709 CPR7L3 44133672 Ki = 71 nM T78709 CE3SD9 44133859 Ki = 37 nM T78709 CZ2VQ1 44133861 Ki = 37 nM T78709 C9P5XU 44133863 Ki = 5.5 nM T78709 C2G7AO 44134036 Ki = 10 nM T78709 C5YKI9 44134038 Ki = 11 nM T78709 C6DQJ3 44134039 Ki = 7.2 nM T78709 C8RZX0 44134041 Ki = 173 nM T78709 CXZH39 44138098 Ki = 0.2512 nM T78709 CUOD42 44138104 Ki = 0.1585 nM T78709 C8R1QU 44178224 Ki = 12.4 nM T78709 CW3X1D 44182545 Ki = 2.81 nM T78709 CI8SO3 44182695 Ki = 71.9 nM T78709 CQP5G0 44182696 Ki = 7.72 nM T78709 CYMQ43 44182839 Ki = 44.3 nM T78709 C6SG0O 44192200 Ki = 3.7 nM T78709 CMR7T1 44204999 EC50 = 50.12 nM T78709 CVG6X1 44209472 Ki = 3.6 nM T78709 CD5AB7 44209480 Ki = 1.1 nM T78709 CXR6K7 44212701 Ki = 6.5 nM T78709 C8ORL9 44212702 Ki = 9.2 nM T78709 CN71EI 44212703 Ki = 12 nM T78709 CSK83C 44213966 IC50 = 3.981 nM T78709 C69CVF 44213967 IC50 = 25.12 nM T78709 C34HLC 44213968 IC50 = 5.012 nM T78709 C8EDC7 44214579 Ki = 36.4 nM T78709 CIHS31 44219920 Ki = 20 nM T78709 CL0SN8 44219921 Ki = 32.9 nM T78709 C36ZRH 44219922 Ki = 17.2 nM T78709 CHY51E 44219923 Ki = 7.2 nM T78709 CC4RT6 44220111 Ki = 172 nM T78709 CL12NI 44220112 Ki = 47.3 nM T78709 C21PGV 44220113 Ki = 167 nM T78709 C4QOE7 44220114 Ki = 5.5 nM T78709 CTK38P 44220115 Ki = 2.8 nM T78709 C2M9DC 44220314 Ki = 6.8 nM T78709 C8I4KR 44220315 Ki = 2 nM T78709 CVW0O8 44220316 Ki = 1.5 nM T78709 C2FDB1 44250364 IC50 > 10000 nM T78709 C8MC0Q 44251387 IC50 > 10000 nM T78709 C5YEA8 44251388 IC50 > 10000 nM T78709 C0BSF6 44251389 IC50 > 10000 nM T78709 C2K0VZ 44253016 EC50 > 3162.28 nM T78709 CL09IQ 44263496 IC50 > 10000 nM T78709 C87MXH 44263497 IC50 > 10000 nM T78709 CT8MG3 44266611 Ki = 317 nM T78709 CFQ4L9 44266612 Ki = 338 nM T78709 C4QVN3 44266613 Ki = 49 nM T78709 C7AWM2 44266623 Ki = 10 nM T78709 CZ36NP 44266636 Ki = 16 nM T78709 CK0XI3 44266651 Ki = 4.9 nM T78709 CP52AC 44266663 Ki > 1000 nM T78709 C5RH3X 44266664 Ki < 1 nM T78709 C2Q4YJ 44266668 Ki = 16 nM T78709 CS6F3H 44266676 Ki = 1 nM T78709 CIO03X 44266677 Ki = 54 nM T78709 CW14OJ 44266678 Ki > 442 nM T78709 CN90JC 44266689 Ki = 252 nM T78709 CB2RF4 44266863 Ki = 4.5 nM T78709 CCP37Q 44267158 IC50 = 3019.95 nM T78709 CFEI56 44267161 IC50 = 512.86 nM T78709 CHU4L9 44267168 IC50 = 15848.93 nM T78709 CIZ5W7 44267181 IC50 = 234.42 nM T78709 CFE12G 44267205 IC50 = 15848.93 nM T78709 C5CPZ7 44267215 IC50 = 4168.69 nM T78709 CO65VL 44269006 Ki = 70.79 nM T78709 C0TP2Z 44269013 Ki = 79.43 nM T78709 CWR1Q3 44269487 Ki > 1000 nM T78709 CZ0YI5 44269492 Ki = 7 nM T78709 CLY2H7 44269511 Ki > 1000 nM T78709 C9QK2C 44269512 Ki = 611 nM T78709 CV0S8B 44269559 Ki = 12 nM T78709 CDC0H2 44269581 Ki = 28 nM T78709 C46WGB 44269582 Ki = 93 nM T78709 CE8NI2 44269606 Ki = 247 nM T78709 CGA1W5 44269820 Ki = 2000 nM T78709 C0C4QN 44269825 Ki = 1500 nM T78709 CIN1S4 44272400 IC50 = 4.571 nM T78709 C13QRS 44272402 IC50 = 72.44 nM T78709 CJ15FQ 44272419 IC50 = 9.12 nM T78709 CQ83VT 44274687 Ki = 2.2 nM T78709 C4MHT3 44274739 Ki = 470 nM T78709 CEY19W 44274740 Ki = 0.2 nM T78709 CD2KU5 44274871 Ki = 16 nM T78709 CNDU40 44274872 Ki = 1 nM T78709 C6U4TV 44274892 Ki = 1000 nM T78709 CC38DG 44274893 Ki = 317 nM T78709 CN01UL 44274899 Ki = 0.1 nM T78709 CLG10Y 44275015 Ki > 470 nM T78709 CU4KC2 44275016 Ki = 0.2 nM T78709 CBG61X 44275031 Ki = 236 nM T78709 C5SBH4 44275061 Ki = 1000 nM T78709 CSY7E4 44275135 Ki = 62 nM T78709 CVUE38 44275155 Ki = 54 nM T78709 CH3V9B 44275206 Ki = 442 nM T78709 CIRX69 44275207 Ki = 54 nM T78709 C86EDH 44275362 Ki = 105 nM T78709 CBV7O8 44275604 Ki = 6.4 nM T78709 CQ19YR 44275615 Ki = 304 nM T78709 CE60XZ 44275616 Ki = 80 nM T78709 C6JI7M 44275657 Ki = 104 nM T78709 CFA79L 44275658 Ki = 11 nM T78709 C1H0XC 44275766 Ki = 5.4 nM T78709 CNHE76 44276598 Ki = 170 nM T78709 CC2OD4 44278111 Ki > 10000 nM T78709 CRMA84 44278114 Ki > 10000 nM T78709 CF0Y4M 44278115 Ki = 3967.7 nM T78709 C08LZS 44279525 Ki = 0.96 nM T78709 C1OI7G 44279549 Ki = 5.8 nM T78709 CFWE96 44279550 Ki = 4 nM T78709 C7DR8P 44279889 Ki = 14 nM T78709 C51NLQ 44289248 Ki = 15.14 nM T78709 CWC49F 44289261 Ki = 6.31 nM T78709 C1JX5M 44289437 Ki = 10.96 nM T78709 CIM92E 44289525 Ki = 11.75 nM T78709 COQ53S 44290346 EC50 = 47.86 nM T78709 CU1S5W 44292309 IC50 = 46 nM T78709 C2C4UE 44292323 IC50 = 930 nM T78709 CM25WH 44292490 IC50 = 4 nM T78709 CGM6S1 44292505 IC50 = 710 nM T78709 C35JVN 44292507 IC50 = 840 nM T78709 CNKH68 44292523 IC50 = 64 nM T78709 C4KX1F 44292555 IC50 = 99 nM T78709 CM6A3I 44292629 IC50 = 460 nM T78709 CB0CD4 44292676 IC50 = 69 nM T78709 CLZ25G 44292706 IC50 = 210 nM T78709 C68SAH 44292707 IC50 = 1460 nM T78709 C0XYU8 44292776 IC50 = 87 nM T78709 CJK5G1 44292790 IC50 > 1000 nM T78709 CNQ82Z 44294182 Ki < 1000 nM T78709 C1IWT4 44296810 IC50 = 489.78 nM T78709 C8BXD4 44299396 Ki = 9.12 nM T78709 CV3PH7 44299504 Ki = 4.83 nM T78709 C0OX9M 44299511 Ki = 9.31 nM T78709 C59XUA 44299512 Ki = 29.4 nM T78709 C7U4DQ 44299513 Ki = 6.79 nM T78709 CJ0EQ1 44299524 Ki = 5.17 nM T78709 CWL48T 44299539 Ki = 7.64 nM T78709 C3QE4F 44299553 Ki = 6.07 nM T78709 CSTJ48 44299556 Ki = 7.21 nM T78709 COK1E4 44299569 Ki = 15.35 nM T78709 C14YCS 44299581 Ki = 7.5 nM T78709 CT48UN 44299643 Ki = 7.45 nM T78709 C2X0BS 44299664 Ki = 3.13 nM T78709 C0VXZ9 44299672 Ki = 1.44 nM T78709 CO6MJ9 44299681 Ki = 6.13 nM T78709 C2U0XO 44299682 Ki = 19.85 nM T78709 COCL75 44299716 Ki = 7.12 nM T78709 COI7M3 44299729 Ki = 1.89 nM T78709 C9K5QI 44299730 Ki = 4.7 nM T78709 CHZ3J7 44299764 Ki = 451.6 nM T78709 CH19QL 44299885 Ki = 14.15 nM T78709 CHD2X3 44299886 Ki = 27.83 nM T78709 C6T9BK 44299887 Ki = 22.6 nM T78709 CXYI48 44299888 Ki = 10.4 nM T78709 C9GX3Z 44299892 Ki = 12.66 nM T78709 CT74SG 44299914 Ki = 6.28 nM T78709 C89HGM 44299915 Ki = 3.09 nM T78709 CM8KV2 44300018 Ki = 4.24 nM T78709 CBSQ04 44300865 Ki = 790 nM T78709 CQ5A2E 44301054 Ki = 450 nM T78709 CEF72W 44305547 IC50 = 7762.47 nM T78709 CW07BA 44306007 IC50 = 457088.19 nM T78709 CKY68S 44309775 Ki = 941 nM T78709 C1TKV6 44309876 Ki = 540 nM T78709 C3L1OJ 44310701 Ki = 17 nM T78709 C8JP5T 44315098 Ki = 200 nM T78709 CN9ZV0 44315099 Ki = 17 nM T78709 C9BTW3 44315120 Ki = 130 nM T78709 CFB13Y 44315131 Ki = 41 nM T78709 CYVZ78 44315380 Ki = 32 nM T78709 C6AWP3 44315381 Ki = 26 nM T78709 C83WGQ 44315382 Ki = 49 nM T78709 CP9D6G 44315383 Ki = 85 nM T78709 CV4X1P 44315386 Ki = 15 nM T78709 C9G2KL 44315406 Ki = 7.6 nM T78709 C2HUA3 44315407 Ki = 21 nM T78709 CHJ1I7 44315426 Ki = 42 nM T78709 CFE15Q 44315427 Ki = 14 nM T78709 C8S5RH 44315436 Ki = 32 nM T78709 CL0Z3J 44315453 Ki = 23 nM T78709 CF3VK8 44315548 Ki = 7.9 nM T78709 C49OQD 44315568 Ki = 38 nM T78709 C7TCE9 44315569 Ki = 35 nM T78709 C1P0XE 44316740 Ki = 8.37 nM T78709 C62EYI 44316755 Ki = 14.45 nM T78709 CVKF37 44316789 Ki = 1.8 nM T78709 CFK6D0 44316790 Ki = 2.33 nM T78709 CGX14Y 44316815 Ki = 11.66 nM T78709 C2GKY9 44316828 Ki = 24.23 nM T78709 COM46U 44316963 Ki = 6.85 nM T78709 C65CRT 44316964 Ki = 0.98 nM T78709 C4M6VT 44316965 Ki = 11.75 nM T78709 C9TXA5 44316966 Ki = 16.48 nM T78709 C2PB8C 44317057 Ki = 2.98 nM T78709 C18BYV 44317081 Ki = 1.76 nM T78709 CLZH14 44317082 Ki = 5.67 nM T78709 CFY17P 44317084 Ki = 15.7 nM T78709 CXOP69 44317095 Ki = 5.26 nM T78709 C6E4UA 44317120 Ki = 4.23 nM T78709 CL78IT 44317121 Ki = 5.52 nM T78709 CTK8U7 44317134 Ki = 4.88 nM T78709 CBMS83 44317146 Ki = 3.09 nM T78709 C9Y4LX 44317147 Ki = 94.9 nM T78709 CV8WZ0 44318454 IC50 = 1584.89 nM T78709 CXJL56 44318842 IC50 > 1000 nM T78709 CHT83A 44320347 Ki = 3 nM T78709 C02LRC 44322770 Ki = 3.7 nM T78709 C40NAS 44322821 IC50 = 19.95 nM T78709 CZ7JF6 44322823 IC50 = 50.12 nM T78709 CSQT84 44322859 IC50 > 100 nM T78709 CR0DQ4 44322885 IC50 = 15.85 nM T78709 C5WL1J 44322886 IC50 = 1.585 nM T78709 C37UTX 44322916 IC50 = 1.995 nM T78709 C3C1OY 44322934 IC50 = 12.59 nM T78709 CJC37P 44322940 IC50 > 1000 nM T78709 C2LV3J 44322952 IC50 > 1000 nM T78709 C1MTR2 44322963 IC50 > 1000 nM T78709 C5R2NL 44322965 IC50 > 1000 nM T78709 C5UFN9 44323074 IC50 = 7.943 nM T78709 CTE2Y6 44323104 Ki = 1.84 nM T78709 CW2P4D 44323130 Ki = 1.43 nM T78709 CQ4C8I 44323137 Ki = 1.39 nM T78709 C3CZF1 44323147 IC50 = 7.943 nM T78709 CEH78W 44323156 IC50 = 125.89 nM T78709 CW7F6I 44323157 IC50 = 50.12 nM T78709 CLN5S4 44323161 IC50 = 15.85 nM T78709 CQI51B 44323162 IC50 = 5.012 nM T78709 CHG3F0 44323163 IC50 > 1000 nM T78709 CPB3U4 44323179 Ki = 1.82 nM T78709 CR14CB 44323200 IC50 > 1000 nM T78709 C9LUP6 44323231 IC50 = 3.981 nM T78709 CD26JI 44323253 IC50 = 1.259 nM T78709 CE7B0T 44323254 IC50 = 12.59 nM T78709 CE8VP0 44323267 IC50 > 1000 nM T78709 CW16JD 44324737 Ki > 1000 nM T78709 CA84SN 44324765 Ki > 1000 nM T78709 COA3H4 44324800 Ki = 475 nM T78709 CY04JW 44324972 Ki > 1000 nM T78709 CV56DM 44326256 Ki = 120 nM T78709 CV8A2N 44326257 Ki = 7.8 nM T78709 C2X9GN 44326324 Ki = 3.9 nM T78709 C2YZI8 44334603 Ki = 0.6 nM T78709 C1DH4T 44334637 Ki = 0.4 nM T78709 C6BJZ0 44335519 Ki = 92.6 nM T78709 C5JCR2 44335674 Ki = 19.6 nM T78709 CLG1Q8 44336170 EC50 = 0.78 nM T78709 C01UJW 44336554 EC50 > 100000 nM T78709 CS7NA2 44337678 Ki = 8 nM T78709 CU4F3W 44337731 Ki > 1000 nM T78709 CUT24A 44338900 Ki = 405 nM T78709 C03OMP 44342812 Ki = 6.7 nM T78709 C2VD8T 44342867 Ki = 32.9 nM T78709 CQ39UH 44342906 Ki = 45.4 nM T78709 C1LID6 44343052 Ki = 142 nM T78709 C7MLO1 44343055 Ki = 15.7 nM T78709 CMLA57 44343195 Ki = 391 nM T78709 CEA06L 44343196 Ki = 156 nM T78709 CD62CF 44345026 Ki = 860 nM T78709 C6N3XK 44345317 IC50 < 1000 nM T78709 CCU89V 44350664 Ki = 414.4 nM T78709 CJ14XP 44351290 Ki = 13.48 nM T78709 C2RU7Y 44351301 Ki = 9.42 nM T78709 CK0ME4 44351312 Ki = 9.2 nM T78709 C6NQ0M 44351330 Ki = 26.77 nM T78709 CT6Q4O 44351331 Ki = 4.06 nM T78709 C4Y6QD 44351334 Ki = 12.65 nM T78709 CHGF01 44351335 Ki = 12.35 nM T78709 CJX4D0 44351341 Ki = 23.15 nM T78709 CQ28XE 44351344 Ki = 15.65 nM T78709 C03RQI 44351345 Ki = 5.65 nM T78709 C43ZES 44351406 Ki = 7.11 nM T78709 C9Y8IW 44351426 Ki = 2.12 nM T78709 C5PZ7I 44351452 Ki = 20.2 nM T78709 CO5G7D 44351470 Ki = 14.35 nM T78709 CD0SK8 44351501 Ki = 10.52 nM T78709 C95TIX 44351508 Ki = 4.84 nM T78709 CZD3O8 44351509 Ki = 6.36 nM T78709 CS51MO 44351512 Ki = 28.1 nM T78709 C2D1RC 44351513 Ki = 19.38 nM T78709 CJ2ZT4 44351521 Ki = 104.63 nM T78709 CHGY49 44351527 Ki = 32 nM T78709 CIK31Q 44351535 Ki = 9.8 nM T78709 CX3ZL5 44351656 Ki = 71.7 nM T78709 CUXH48 44352308 Ki = 265 nM T78709 CH9F8G 44356232 Ki = 218.78 nM T78709 C3I9DE 44358574 Ki = 0.23 nM T78709 CJ80OW 44360984 Ki = 11 nM T78709 CS8K1A 44360992 Ki = 22 nM T78709 C3NZ7B 44361021 Ki = 15 nM T78709 CS3J6N 44363580 Ki > 100 nM T78709 C3LKN1 44364048 Ki = 1.995 nM T78709 C2MZ6D 44365404 Ki = 3.05 nM T78709 CSTQ01 44365426 Ki = 39 nM T78709 CFO5K8 44365439 Ki = 0.33 nM T78709 CV54RI 44365467 Ki = 16.7 nM T78709 CO4I2K 44365657 Ki = 5.87 nM T78709 CB0A1W 44365671 Ki = 0.81 nM T78709 C4AWE7 44365672 Ki = 1.53 nM T78709 C0RLY6 44365679 Ki = 1.6 nM T78709 CH26LQ 44365682 Ki = 127.7 nM T78709 CTE15U 44365700 Ki = 2.92 nM T78709 C40CAM 44365701 Ki = 61.6 nM T78709 C1M0OB 44365720 Ki = 307.1 nM T78709 CVU16E 44365728 Ki = 46 nM T78709 C10HST 44365811 Ki = 357 nM T78709 CPV96F 44367514 Ki = 1.5 nM T78709 C6CJ7S 44373641 Ki = 9.8 nM T78709 C1YIJ4 44373989 Ki = 3.8 nM T78709 CVL3U2 44374207 Ki = 41 nM T78709 CQ79MO 44374219 Ki = 11 nM T78709 CV8CP3 44374225 Ki = 2200 nM T78709 C04WKH 44374233 Ki = 37 nM T78709 CB2S7T 44374234 Ki = 1200 nM T78709 CH03ON 44374236 Ki = 7.6 nM T78709 CJ4A2U 44374299 Ki = 210 nM T78709 CD9QP8 44374649 Ki > 1786 nM T78709 C4BAI3 44374753 IC50 > 10000 nM T78709 CJ4KP3 44377759 Ki = 74 nM T78709 CE06VB 44377955 Ki = 0.89 nM T78709 C4VXQ1 44388858 Ki = 41 nM T78709 CTPG47 44388956 Ki = 115 nM T78709 CQ85AW 44389003 Ki > 2000 nM T78709 C8AG7U 44389016 Ki = 875 nM T78709 CV14HS 44389135 Ki = 194 nM T78709 CTZ7P5 44389374 Ki < 100 nM T78709 CC6XK1 44389508 Ki = 107.15 nM T78709 C6U3FH 44389522 Ki = 46.77 nM T78709 C74BRC 44389523 Ki = 16.6 nM T78709 C7DT6S 44391257 Ki = 0.5012 nM T78709 CV4PR8 44391267 Ki = 2.512 nM T78709 C0UEV5 44391270 Ki = 1.585 nM T78709 CL8G4N 44391284 Ki = 12.59 nM T78709 C35BYM 44391300 Ki = 1.259 nM T78709 C1PT7D 44391314 Ki = 1.585 nM T78709 CLZ83B 44391323 Ki = 1.995 nM T78709 C1XVH3 44391327 Ki = 10 nM T78709 C9P3WI 44391358 Ki = 7.943 nM T78709 C9XF0B 44391374 Ki = 100 nM T78709 CNO6S7 44391393 Ki = 6.31 nM T78709 C53UVJ 44393088 Ki > 100 nM T78709 C6WAK2 44393173 Ki = 87.1 nM T78709 CEO2W9 44393372 Ki = 27 nM T78709 CXP4Q7 44393393 Ki = 24 nM T78709 C6BZS0 44393403 Ki = 33 nM T78709 C86NED 44393411 Ki = 46 nM T78709 C9THO4 44393415 Ki = 10 nM T78709 CYOU64 44395296 Ki = 173.2 nM T78709 CECK89 44395347 Ki = 320 nM T78709 C3RV6T 44395741 Ki = 90.9 nM T78709 CN02LY 44395762 Ki = 240 nM T78709 CLH1T7 44395786 Ki = 160 nM T78709 C9K4SC 44395787 Ki = 310 nM T78709 C93XHA 44395809 Ki = 12 nM T78709 CTA27N 44395810 Ki = 860 nM T78709 C9A4NM 44395832 Ki = 11 nM T78709 C4B0OI 44397588 Ki = 794.33 nM T78709 C5FP0R 44397589 Ki = 1000 nM T78709 CE3G8U 44397670 Ki = 501.19 nM T78709 C1KA3F 44400359 Ki = 63.1 nM T78709 C0E5HY 44400500 Ki = 12 nM T78709 CO8EU5 44400519 Ki = 77 nM T78709 CRX12E 44400553 Ki = 14 nM T78709 CIU18E 44400585 Ki = 20 nM T78709 CV8K2W 44400594 Ki = 210 nM T78709 C84RNU 44400626 Ki = 27 nM T78709 CY94SF 44400674 Ki = 0.5 nM T78709 C9THQ3 44402868 Ki = 501.19 nM T78709 C1EI5Q 44402869 Ki = 79.43 nM T78709 CV0PC9 44402870 Ki = 50.12 nM T78709 CV15IH 44402871 Ki = 1584.89 nM T78709 CG1WU9 44402876 Ki = 12.59 nM T78709 C6WNI4 44402877 Ki = 501.19 nM T78709 CDL1F6 44402878 Ki = 1000 nM T78709 C1B4QL 44403095 Ki = 52.5 nM T78709 C1YL7Z 44403098 Ki = 1079 nM T78709 CFV98A 44403101 Ki = 405 nM T78709 C6OY9S 44403102 Ki = 382 nM T78709 CH4SX6 44403105 Ki = 882 nM T78709 C12FIH 44403106 Ki = 15.4 nM T78709 CQ4U2P 44403210 Ki = 15 nM T78709 CKE6T4 44403213 Ki = 60 nM T78709 CAJX39 44403214 Ki = 22 nM T78709 C61CNS 44403219 Ki = 28 nM T78709 C5AE9L 44403220 Ki = 24 nM T78709 CC6XM4 44403224 Ki = 30 nM T78709 C6JB4M 44403225 Ki = 51 nM T78709 CGE52H 44403232 Ki = 120 nM T78709 CI0WG5 44404225 Ki = 0.7943 nM T78709 C7FAW3 44404229 Ki = 1 nM T78709 C0MXR4 44404230 Ki = 10 nM T78709 C7OD6Q 44404236 Ki = 5.012 nM T78709 C5W2KR 44404240 Ki = 3.162 nM T78709 CI50CY 44404241 Ki = 3.981 nM T78709 CF69DU 44404244 Ki = 5.012 nM T78709 CE0NI6 44404245 Ki = 6.31 nM T78709 CLW3P7 44404249 Ki = 0.3162 nM T78709 CF8LN5 44404253 Ki = 1.259 nM T78709 C3LI6E 44404258 Ki = 3.162 nM T78709 C2NH8G 44404260 Ki = 6.31 nM T78709 C7R5HU 44404264 Ki = 31.62 nM T78709 CVTZ13 44404268 Ki = 1.585 nM T78709 C18ISW 44404272 Ki = 1.259 nM T78709 C4LKC1 44404394 Ki = 335 nM T78709 C3EJ4G 44404396 Ki = 315 nM T78709 C4Q2BS 44404551 Ki = 45 nM T78709 C7W3BP 44405573 Ki = 4.1 nM T78709 CV9IR7 44405574 Ki = 0.9 nM T78709 CFG72V 44405575 Ki = 1.9 nM T78709 C8WSZ2 44405586 Ki = 0.7 nM T78709 CEJ0C3 44405587 Ki = 2.5 nM T78709 C4DK0U 44405655 Ki = 5.6 nM T78709 C28WCH 44405665 Ki = 103.9 nM T78709 CS7ZD5 44405666 Ki = 0.6 nM T78709 CIH9J0 44405669 Ki = 0.4 nM T78709 CVZO38 44405677 Ki = 18.8 nM T78709 CMK32Z 44405701 Ki = 1.5 nM T78709 CZK5L6 44405702 Ki = 0.9 nM T78709 CO7G3W 44405725 Ki = 2.5 nM T78709 CU1VL9 44405726 Ki = 2.5 nM T78709 CO1P3W 44405730 Ki = 0.3 nM T78709 C65PBE 44405930 Ki = 113.4 nM T78709 CBGH16 44405935 Ki = 157.3 nM T78709 CF4S3Y 44405965 Ki = 1540 nM T78709 CT3Z8U 44405980 Ki = 1030 nM T78709 CQ7RI8 44405981 Ki = 19.1 nM T78709 C0BI5F 44405985 Ki = 64.9 nM T78709 C1FZE7 44405991 Ki = 295.1 nM T78709 C4NC8M 44405995 Ki = 1450 nM T78709 CVM1Y5 44406002 Ki = 333.34 nM T78709 C0R5VL 44406003 Ki = 1815 nM T78709 C90NQJ 44406012 Ki = 401.3 nM T78709 CL5C9T 44406077 Ki = 1070 nM T78709 CPNT73 44408681 Ki = 2.81 nM T78709 C81GYD 44408682 Ki = 7.25 nM T78709 C9J2VU 44408685 Ki = 30.21 nM T78709 CH9MC5 44408702 Ki = 12.76 nM T78709 C9IPV4 44408784 Ki = 103 nM T78709 C54EOX 44408852 Ki = 7.14 nM T78709 CCM7A1 44408853 Ki = 75.18 nM T78709 CM41IO 44408882 Ki = 8.15 nM T78709 CEM05A 44408883 Ki = 5.86 nM T78709 C5CKA7 44408888 Ki = 8.46 nM T78709 CUM50D 44408890 Ki = 6.91 nM T78709 C9R2BF 44408942 Ki = 15.31 nM T78709 CU15IW 44408946 Ki = 10.98 nM T78709 CG87PW 44409290 Ki > 720 nM T78709 CO4SX2 44412809 Ki = 230 nM T78709 C05FOC 44412810 Ki = 260 nM T78709 CILZ93 44412825 Ki = 63 nM T78709 CB1TC6 44412826 Ki = 69 nM T78709 C32NFQ 44412838 Ki = 40 nM T78709 CR5D1B 44412906 Ki = 40 nM T78709 C95HRZ 44412907 Ki = 480 nM T78709 CN02QD 44412913 Ki = 25 nM T78709 CHRS85 44412928 Ki = 170 nM T78709 CWD97B 44412932 Ki = 17 nM T78709 CC7Y5W 44412934 Ki = 24 nM T78709 COJ75S 44412935 Ki = 11 nM T78709 C9LS4E 44412965 Ki = 12 nM T78709 CS1GP5 44412966 Ki = 27 nM T78709 CFKI28 44412969 Ki = 4 nM T78709 CVDM51 44412991 Ki = 12 nM T78709 CHW6K9 44413006 Ki = 17 nM T78709 CFY4W8 44413015 Ki = 50 nM T78709 CAJI08 44413016 Ki = 17 nM T78709 CV8SQ0 44413025 Ki = 18 nM T78709 CC0UA4 44413026 Ki = 9 nM T78709 CR4Z8C 44413037 Ki = 15 nM T78709 CJN6P4 44427818 Ki = 6.71 nM T78709 CW3F5H 44427820 Ki = 29.7 nM T78709 CYLO03 44427821 Ki = 309 nM T78709 CJY9L5 44427822 Ki = 92 nM T78709 CO46HS 44427823 Ki = 60.6 nM T78709 CFG0S3 44427824 Ki = 666 nM T78709 C7PK0M 44427825 Ki = 21.7 nM T78709 CDV6A3 44427826 Ki = 71.8 nM T78709 C65ZXC 44427827 Ki = 34.3 nM T78709 CZ0X7U 44427829 Ki = 1810 nM T78709 C9U8YT 44427831 Ki = 36.2 nM T78709 C0C8AH 44427835 Ki = 117 nM T78709 C8EV3G 44427836 Ki = 15.1 nM T78709 CS9ND5 44427841 Ki = 59 nM T78709 COV6N3 44427842 Ki = 982 nM T78709 C6JK5A 44431532 Ki = 115 nM T78709 C5LNH6 44431533 Ki = 105 nM T78709 CLX73C 44431534 Ki = 307 nM T78709 C4P5XG 44431536 Ki = 26 nM T78709 CYPR70 44431537 Ki = 16 nM T78709 CVX7A6 44433249 Ki = 40.6 nM T78709 C5P4OW 44433250 Ki = 3.89 nM T78709 C3YV6I 44433251 Ki = 11.2 nM T78709 C0AT6Q 44433252 Ki = 26.1 nM T78709 C1SK2A 44433253 Ki = 18.3 nM T78709 COH61M 44433254 Ki = 1450 nM T78709 CPO7H6 44433255 Ki = 868 nM T78709 C8YPF6 44433257 Ki = 872 nM T78709 CZLT14 44433258 Ki = 125 nM T78709 CP0F4L 44433280 Ki > 3000 nM T78709 C4TN2F 44433281 Ki = 833 nM T78709 C6W8GQ 44433303 Ki = 76.1 nM T78709 CZK39E 44437329 Ki = 1.7 nM T78709 CKZF16 44439165 Ki = 2.512 nM T78709 CA4HZ3 44439167 Ki = 10 nM T78709 CT0C4I 44443093 Ki = 1.585 nM T78709 C8E1AC 44443094 Ki = 1.259 nM T78709 CZ6BK9 44443095 Ki = 0.2512 nM T78709 CV5T2C 44443096 Ki = 1.259 nM T78709 CT1S6L 44443097 Ki = 1.995 nM T78709 CF1V8O 44443098 Ki = 3.981 nM T78709 CHZ48Q 44443101 Ki = 1.259 nM T78709 CQ53TV 44443130 Ki = 7.943 nM T78709 CEZ6U8 44443131 Ki = 3.162 nM T78709 CN4XZ6 44443132 Ki = 2.512 nM T78709 C5RVE0 44446999 Ki = 4.9 nM T78709 C9E0FL 44447001 Ki = 2 nM T78709 CSJ4U5 44447002 Ki = 5 nM T78709 CL87PU 44447003 Ki = 5.5 nM T78709 CCD6B5 44447005 Ki = 12 nM T78709 CBH65G 44447007 Ki = 12 nM T78709 C8CF7X 44447008 Ki = 41.8 nM T78709 CN3EH7 44447010 Ki = 28.1 nM T78709 CYWP06 44447012 Ki = 56 nM T78709 C41KNM 44447013 Ki = 66.7 nM T78709 CE12BC 44447015 Ki = 4.5 nM T78709 CUD31L 44447018 Ki = 20.9 nM T78709 CNLX79 44447028 Ki = 37.2 nM T78709 CM8K1H 44447039 Ki = 7.9 nM T78709 C5IJW2 44447059 Ki = 6.5 nM T78709 CHXF10 44447061 Ki = 1 nM T78709 CG93OH 44447063 Ki = 2 nM T78709 C9KJR2 44447065 Ki = 2 nM T78709 C5QK8Z 44447067 Ki = 2 nM T78709 C7A6RP 44447068 Ki = 1 nM T78709 CM8P9A 44447070 Ki = 7.8 nM T78709 CK4HA6 44447072 Ki = 7.7 nM T78709 C2S6HQ 44448054 Ki = 373 nM T78709 C3Z7FI 44451927 IC50 = 960 nM T78709 C57SBC 44451980 IC50 = 120 nM T78709 CEST18 44451982 IC50 = 220 nM T78709 CRN4F8 44452007 IC50 = 370 nM T78709 CG1C6X 44452142 IC50 = 140 nM T78709 CVAU93 44452222 IC50 = 500 nM T78709 C0B3LC 44452327 IC50 = 400 nM T78709 CZL97F 44455426 Ki > 10000 nM T78709 CYS7T4 44455943 Ki = 765 nM T78709 C6BFI0 44456033 Ki = 95.2 nM T78709 CG91RD 44456395 Ki = 339 nM T78709 C12XGE 44456400 Ki > 10000 nM T78709 CZ1BM3 44461160 EC50 = 251.19 nM T78709 CD5L8N 44461162 EC50 = 12.59 nM T78709 CQ2IX7 44461606 IC50 > 1000 nM T78709 C4DL5C 44469677 IC50 = 1 nM T78709 CM5EY8 44474470 IC50 > 1000 nM T78709 C8UON6 44474625 IC50 > 1000 nM T78709 C6HVU1 44474629 IC50 > 10000 nM T78709 CE2Z8S 44474631 IC50 > 10000 nM T78709 C8LA4W 44474797 IC50 > 1000 nM T78709 CJ10OZ 44531812 Ki = 3090 nM T78709 C4SX7H 44537919 Ki = 105 nM T78709 CVD14L 44537925 Ki = 133 nM T78709 C3D4HR 44537940 Ki > 5000 nM T78709 CT85QK 44538690 Ki = 1330 nM T78709 C4LUK7 44549156 Ki = 7.244 nM T78709 CJ7U3K 44554227 Ki > 5000 nM T78709 CM0I1P 44554393 Ki > 5000 nM T78709 CNHA47 44554395 Ki = 1780 nM T78709 C6WV2P 44559406 IC50 > 10000 nM T78709 CB23PH 44560995 Ki = 19 nM T78709 C0N1LV 44561105 IC50 = 2.3 nM T78709 C7MAT0 44568331 Ki = 1.7 nM T78709 CVA67X 44568347 Ki = 450 nM T78709 CQF70H 44568357 Ki = 3 nM T78709 C6LK9P 44568358 Ki = 3.6 nM T78709 CIB94E 44568385 Ki = 8.3 nM T78709 COE94C 44568461 Ki = 9.1 nM T78709 CI0F2C 44568462 Ki = 42.6 nM T78709 CAR23X 44568818 Ki = 37.15 nM T78709 CAO31F 44568917 Ki = 7.586 nM T78709 CE3GV8 44568918 Ki = 229.09 nM T78709 C9LP7Z 44575219 EC50 = 9000 nM T78709 CZO5Y8 44580740 Ki = 3.162 nM T78709 C4N6PM 44580741 Ki = 1.585 nM T78709 C0XVL5 44580783 Ki = 125.89 nM T78709 C4SD7P 44580784 Ki = 0.2512 nM T78709 CNOU35 44581235 Ki = 7.943 nM T78709 CO6E5K 44581260 Ki = 5.012 nM T78709 CS6HG9 44581603 Ki = 6.31 nM T78709 C1HAQ2 44581604 Ki = 12.59 nM T78709 CRCH48 44582675 Ki > 10000 nM T78709 CEJ4R8 44582676 Ki = 1681 nM T78709 CZGP86 44582677 Ki > 10000 nM T78709 C5QB4K 44582678 Ki > 10000 nM T78709 C01RCI 44582705 Ki = 1883 nM T78709 CXL25V 44582706 Ki > 10000 nM T78709 C8MR1X 44582707 Ki = 1723 nM T78709 C4IT1N 44582708 Ki = 991 nM T78709 CSF39B 44588698 Ki = 630.96 nM T78709 C60NYB 44588704 Ki = 0.66 nM T78709 C7SKM1 44588720 Ki = 398.11 nM T78709 CI6SO1 44588721 Ki = 50.12 nM T78709 CB14UQ 44588722 Ki = 79.43 nM T78709 CNK64D 44588742 Ki = 158.49 nM T78709 CAT73D 44588743 Ki > 10000 nM T78709 C6DK3E 44588744 Ki > 1584.89 nM T78709 C9BO7K 44588745 Ki = 316.23 nM T78709 CD2CU8 44588771 Ki > 10000 nM T78709 CDIQ25 44588772 Ki = 501.19 nM T78709 CB27TM 44589076 Ki = 0.93 nM T78709 C34YST 44591228 Ki = 75.3 nM T78709 CKV67Q 44591229 Ki = 21.3 nM T78709 C6A2QJ 44591230 Ki = 7.4 nM T78709 CZKV93 44591244 Ki = 32 nM T78709 C1U2NH 44591245 Ki = 5.2 nM T78709 CF20JZ 44591246 Ki = 23.6 nM T78709 CB7QV5 44591259 Ki = 10.4 nM T78709 CQS54L 44591260 Ki = 26.6 nM T78709 CM72EB 44591261 Ki = 35.1 nM T78709 CS56IQ 44591262 Ki = 64.5 nM T78709 C5WRT1 44591263 Ki = 37.8 nM T78709 C1T0XN 44591280 Ki = 38.5 nM T78709 CIGM43 44591281 Ki = 42.5 nM T78709 C1EAR6 44591282 Ki = 40.2 nM T78709 C5E7HO 44591283 Ki = 3420 nM T78709 CZUX15 44591284 Ki = 780 nM T78709 C4VI7E 44591316 Ki = 4450 nM T78709 C3B0GO 44591317 EC50 = 51.4 nM T78709 CW9YA7 44591318 EC50 = 65 nM T78709 CK7XJ0 44591319 EC50 = 40.7 nM T78709 CB0S4Z 44592109 IC50 = 5248.07 nM T78709 C4EH6O 44592207 Ki = 0.2512 nM T78709 CZ5I1N 44592208 Ki > 3162.28 nM T78709 CKM8T7 44592209 Ki = 0.1259 nM T78709 CDJ32U 44592249 Ki = 0.631 nM T78709 CS2FL4 44592250 Ki = 0.1 nM T78709 CL17WU 44592251 Ki = 0.631 nM T78709 CJCL64 44592252 Ki = 0.5012 nM T78709 CM0I3E 44592294 Ki = 0.3162 nM T78709 CQ04EG 44592295 Ki = 0.3981 nM T78709 C65XQL 44592296 Ki = 0.1995 nM T78709 CEB2S1 44592297 Ki = 0.1995 nM T78709 CP51QS 44592332 Ki = 1.585 nM T78709 CD2Z4J 44592333 Ki = 1.995 nM T78709 C7NCT2 44592334 Ki = 6.31 nM T78709 CHY20X 44592335 Ki = 1.585 nM T78709 C5H7XK 44592371 Ki = 3.162 nM T78709 CR8T7B 44593415 Ki = 2.8 nM T78709 C1SN7Y 44593709 Ki = 0.25 nM T78709 CZ0W1I 44593711 Ki = 50.12 nM T78709 CHD0R7 44593712 Ki = 1.98 nM T78709 CPK6N9 44593714 Ki = 1.73 nM T78709 C5HSO3 44593715 Ki = 31.4 nM T78709 CAXK49 44593716 Ki = 7.34 nM T78709 C4WBK1 44593717 Ki = 9.48 nM T78709 CF4Q5M 44593729 Ki = 11.2 nM T78709 C4Y6SW 44598639 Ki = 44 nM T78709 CE9NU2 44598680 Ki = 116 nM T78709 C40ZMK 44598681 Ki = 6.8 nM T78709 CO7K4W 44598682 Ki = 0.67 nM T78709 C96QRP 44598683 Ki = 15 nM T78709 C62CAY 44598684 Ki = 0.47 nM T78709 C52QLW 44598685 Ki = 0.5 nM T78709 C5S3IT 44598725 Ki = 7.8 nM T78709 CXK8A2 44598726 Ki = 73 nM T78709 C0LS9C 44598727 Ki = 29 nM T78709 CL1J3B 44598728 Ki = 54 nM T78709 C67KZG 44608359 EC50 > 10000 nM T78709 CW0RU3 45102635 Ki = 1 nM T78709 C0DLU3 45109862 IC50 = 117 nM T78709 CGB2Z0 45113400 Ki = 7 nM T78709 CMJ1U7 45266443 EC50 > 100000 nM T78709 CEK5G3 45277221 Ki = 63.3 nM T78709 CL3I7B 45277224 Ki = 27 nM T78709 CI4O0A 45277387 Ki = 27.3 nM T78709 CHZ70D 45277559 Ki = 3.76 nM T78709 CZ71RN 45278805 IC50 = 54 nM T78709 CZN6M7 45278882 IC50 = 94 nM T78709 CC86HS 45481874 Ki = 799 nM T78709 C7MO3G 45481875 Ki = 85 nM T78709 CP4OS2 45481876 Ki = 98 nM T78709 CRL6D2 45481877 Ki = 648 nM T78709 C7S9HJ 45481888 Ki = 133 nM T78709 C0HPW1 45481889 Ki = 235 nM T78709 C47HZI 45481890 Ki = 457 nM T78709 CB7SG4 45481891 Ki = 381 nM T78709 C0CHF4 45482789 IC50 = 3600 nM T78709 CZ8G9V 45482876 Ki = 53.7 nM T78709 CX7BE9 45482877 Ki = 204.17 nM T78709 CR80QO 45482879 Ki = 10.96 nM T78709 C9E3JI 45482881 Ki = 100 nM T78709 C1I4FV 45482884 Ki = 416.87 nM T78709 C36LXH 45482890 Ki = 234.42 nM T78709 C6ILK5 45482891 Ki = 398.11 nM T78709 CEOX52 45482892 Ki = 50.12 nM T78709 C1SR9M 45482893 Ki = 30.2 nM T78709 C9LSN3 45482900 Ki = 42.66 nM T78709 C97JBX 45483401 Ki > 4570 nM T78709 C9K4XC 45483416 Ki = 2210 nM T78709 CZQ6H8 45483429 Ki > 1000 nM T78709 C3HAF8 45483430 Ki = 1160 nM T78709 CG2SM9 45483458 Ki = 9 nM T78709 CFM9P8 45483465 Ki = 4 nM T78709 C5DS3M 45483506 Ki = 101 nM T78709 CHCA47 45483511 Ki = 466 nM T78709 C05PBD 46176231 Ki = 66 nM T78709 CI3WX2 46176232 Ki = 279 nM T78709 C4XRY7 46176233 Ki = 35 nM T78709 C4WJ0Z 46176312 Ki = 45 nM T78709 CNW60S 46180190 Ki = 626 nM T78709 C5CET8 46180192 Ki = 12 nM T78709 CEW06P 46180193 Ki = 135 nM T78709 C9PBQ4 46180194 Ki = 6.7 nM T78709 CP8RF4 46180256 Ki = 14 nM T78709 CG8UK9 46180257 Ki = 29 nM T78709 CO7SA6 46180258 Ki = 66 nM T78709 CSY63N 46180259 Ki = 144 nM T78709 C64TDV 46180261 Ki = 373 nM T78709 CQNC52 46180262 Ki > 10000 nM T78709 CBM9O6 46180325 Ki = 149 nM T78709 CP7Y5E 46180326 Ki = 11 nM T78709 C1J3VH 46180327 Ki = 793 nM T78709 CUI5T0 46180329 Ki > 10000 nM T78709 C4Z5LD 46180330 Ki = 340 nM T78709 C73KNC 46180331 Ki = 630 nM T78709 CXQ7G5 46180393 Ki = 90 nM T78709 CHN09F 46180394 Ki = 55 nM T78709 CMS7T5 46180395 Ki = 125 nM T78709 C62FUY 46180396 Ki = 320 nM T78709 C10OKI 46180397 Ki = 510 nM T78709 CM4R8A 46180398 Ki = 3.1 nM T78709 CC7N8T 46180399 IC50 = 18 nM T78709 C62BEZ 46224739 Ki = 19 nM T78709 C34ZXM 46225029 Ki > 10000 nM T78709 C5LTG9 46225164 Ki = 1220 nM T78709 CQT3G4 46225165 Ki = 22 nM T78709 C5OC1A 46225166 Ki = 2 nM T78709 C1AM8J 46225207 Ki = 3 nM T78709 CNQ10M 46225208 Ki = 101 nM T78709 C8Z0DR 46225263 Ki = 85 nM T78709 CYE41P 46225264 EC50 = 22 nM T78709 C2H1PN 46225309 Ki = 4 nM T78709 CUR54A 46225310 Ki = 22 nM T78709 CY82LR 46227396 IC50 > 1000 nM T78709 C06QIT 46227754 EC50 = 25 nM T78709 C30ZIR 46227757 Ki = 23 nM T78709 C4YLZ1 46227762 Ki = 13 nM T78709 C08ZOG 46227770 Ki = 6 nM T78709 CN4HT2 46230756 Ki = 17 nM T78709 CGD6E4 46231118 Ki = 12 nM T78709 CEMB09 46231492 Ki = 12.7 nM T78709 C23JYW 46238348 Ki = 0.79 nM T78709 C42SVX 46700866 IC50 = 1200 nM T78709 CD0K6E 46700867 IC50 = 2100 nM T78709 C5TC2S 46830335 IC50 > 10000 nM T78709 C1K7FL 46830336 IC50 > 10000 nM T78709 C1N4KX 46842383 IC50 > 10000 nM T78709 C0ABR3 46846073 Ki = 2.188 nM T78709 CC62SX 46866711 IC50 = 298 nM T78709 C7ZEI6 46881382 Ki = 0.1288 nM T78709 CN0Q2A 46881443 Ki = 2.63 nM T78709 CGX02N 46881444 Ki = 7.943 nM T78709 C2MC4K 46881463 EC50 = 794.33 nM T78709 CSQ4C9 46881468 EC50 = 3162.28 nM T78709 C4U6RH 46881493 Ki = 8.318 nM T78709 CV7R9S 46881494 Ki = 1.023 nM T78709 C24QFO 46882032 Ki > 1000 nM T78709 C3GQW6 46882033 Ki = 28.84 nM T78709 CPG6U5 46882034 Ki = 1.698 nM T78709 CYB37P 46882085 Ki = 0.8913 nM T78709 CD8CX3 46882086 Ki > 1000 nM T78709 C57GAO 46882087 Ki = 97.72 nM T78709 CV3QW9 46882088 Ki = 7.586 nM T78709 CB8GE1 46884818 IC50 > 10000 nM T78709 C4MQ0A 46884856 IC50 > 10000 nM T78709 CCNT25 46884898 IC50 > 10000 nM T78709 C3MSG2 46885027 IC50 > 10000 nM T78709 CB7XI0 46885213 IC50 > 10000 nM T78709 COH48X 46886853 Ki = 371.54 nM T78709 CBG61I 46886861 Ki = 1445.44 nM T78709 C05KPX 46886862 Ki = 9.333 nM T78709 C1JSH9 46899637 Ki = 0.1259 nM T78709 C3MSL0 46899638 Ki = 0.1585 nM T78709 CV3LP2 46899639 Ki = 0.1259 nM T78709 CGHZ15 46899640 Ki = 0.3981 nM T78709 CN9FC3 46900150 Ki = 0.1259 nM T78709 C40ZJO 46900451 Ki = 0.1995 nM T78709 CNC02A 46900453 Ki = 0.1995 nM T78709 CTCH14 46900455 Ki = 0.1585 nM T78709 CP41AQ 46900457 Ki = 0.1995 nM T78709 CR3L4I 46900459 Ki = 0.07943 nM T78709 CK17PA 46900606 Ki = 0.07943 nM T78709 CQ2K1C 46900608 Ki = 0.5012 nM T78709 C5ZT1B 46900610 Ki = 0.631 nM T78709 C1NAX4 46900612 Ki = 0.3162 nM T78709 CT0SQ2 46900614 Ki = 1.585 nM T78709 CXD9S3 46900776 Ki = 0.1585 nM T78709 C8I7SJ 46900778 Ki = 1 nM T78709 C7QDM9 46900782 Ki = 0.1995 nM T78709 C15FMY 46900954 Ki = 0.1259 nM T78709 C8W1FU 46900956 Ki = 0.1585 nM T78709 CH35BV 46900958 Ki = 0.2512 nM T78709 CA75HK 46914485 Ki = 806 nM T78709 C9D7UW 46914486 Ki = 373 nM T78709 COB4R0 46914487 Ki = 2192 nM T78709 C4JZR8 46914620 Ki = 468 nM T78709 C4JIP7 46914621 Ki = 1720 nM T78709 CZ5TS4 46914771 Ki = 3339 nM T78709 C1LY6Z 46914772 Ki = 3251 nM T78709 C3XE4P 46914773 Ki = 469 nM T78709 C2E6UX 46914774 Ki = 2458 nM T78709 CT36AF 46914775 Ki = 774 nM T78709 CW74CK 46914776 Ki = 4722 nM T78709 CLC27S 46914777 Ki = 3383 nM T78709 CAT12G 46914926 Ki = 599 nM T78709 CE6SQ2 46914927 Ki = 3300 nM T78709 C7FX8L 46931072 Ki = 349 nM T78709 CZDN92 46934426 Ki = 54 nM T78709 C4VG2E 46934427 Ki = 9.62 nM T78709 CUTX67 46934428 IC50 > 1000 nM T78709 CI4XZ1 46934637 Ki = 5.129 nM T78709 CK1Z0M 46934639 Ki = 5.248 nM T78709 CU0TB9 46934641 Ki = 7.244 nM T78709 CR6JV7 46934643 Ki = 5.623 nM T78709 C14ZLO 46934645 Ki = 25.7 nM T78709 C2N9JZ 46934787 Ki = 5.129 nM T78709 CI4U0L 46934789 Ki = 44.67 nM T78709 C8HVG6 46934791 Ki = 3.162 nM T78709 CA51JI 46934793 Ki = 1.259 nM T78709 CB4Z7D 46934945 Ki = 2.63 nM T78709 C6J4TV 46946859 Ki = 0.151 nM T78709 C8V5MJ 46947455 Ki = 2 nM T78709 CY28OS 47556338 Ki = 1551 nM T78709 C4CL9S 49780599 EC50 = 13 nM T78709 C0F4ZA 49780600 EC50 = 8.6 nM T78709 CR61PL 49780603 EC50 = 6.6 nM T78709 CD42FE 49781265 EC50 = 270 nM T78709 C4TP1Q 49781928 EC50 = 52 nM T78709 C2YAD4 49781933 EC50 = 11 nM T78709 CVGW32 49782156 EC50 = 26 nM T78709 C2TGP4 49782388 EC50 = 36 nM T78709 CF2Z7T 49782389 EC50 = 100 nM T78709 C2LZJ0 49783209 Ki = 300 nM T78709 C57SMG 49783415 Ki > 10000 nM T78709 C0TG6I 49783419 Ki > 10000 nM T78709 COE79D 49836152 IC50 = 59.3 nM T78709 C6IN7B 49836154 IC50 > 100 nM T78709 C28CKM 49836301 Ki = 35.48 nM T78709 C5JO6E 49836302 Ki > 10000 nM T78709 C9TNO4 49836303 Ki = 6.026 nM T78709 CR40BA 49836386 IC50 = 1300 nM T78709 C0M5XC 49836496 IC50 = 1100 nM T78709 C8JQ4O 49837354 EC50 = 2.5 nM T78709 CN0MO8 49837461 IC50 < 10 nM T78709 CHB1I9 49837652 IC50 < 10 nM T78709 CG64FA 49837758 IC50 = 96.4 nM T78709 C3OHN0 49850566 Ki = 3.162 nM T78709 C4R2YS 49850567 Ki = 0.5012 nM T78709 CSGQ38 49850568 Ki = 0.7943 nM T78709 C8P5KH 49850569 Ki = 0.3981 nM T78709 C07JTU 49850570 Ki = 1.995 nM T78709 C6FP9W 49850571 Ki = 5.012 nM T78709 C3BVK5 49850668 Ki = 7.943 nM T78709 C6P3RH 49850669 Ki = 3.162 nM T78709 CGYT84 49850670 Ki = 3.981 nM T78709 C6Y3DW 49850671 Ki = 2.512 nM T78709 CK68QR 49850672 Ki = 0.3981 nM T78709 CI6O9A 49850673 Ki = 1.259 nM T78709 COFA76 49850768 Ki = 1.995 nM T78709 C4IX5R 49850769 Ki = 3.162 nM T78709 CXLT59 49850770 Ki = 2.512 nM T78709 C48DOX 49850771 Ki = 3.162 nM T78709 CN5XR1 49850772 Ki = 0.5012 nM T78709 CR4EZ0 49850870 Ki = 0.7943 nM T78709 C5K4EC 49850872 Ki = 1 nM T78709 C8AW0R 49850874 Ki = 1 nM T78709 CB2K6D 49850877 Ki = 0.631 nM T78709 C85KPE 49850980 Ki = 1.259 nM T78709 C5U3YD 49850982 Ki = 2.512 nM T78709 CV62IZ 49850984 Ki = 1.995 nM T78709 CED9V6 49852000 Ki = 1.585 nM T78709 CA0PW5 49852001 Ki = 1.995 nM T78709 C5S6BY 49852002 Ki = 1.995 nM T78709 C13ZTD 49852003 Ki = 6.31 nM T78709 CK17IE 49852105 Ki = 15.85 nM T78709 C6OQV2 49862237 Ki = 103 nM T78709 C6IW4Q 49862238 Ki > 1000 nM T78709 CDHY90 49864027 Ki = 2439 nM T78709 C9KIU1 49864289 IC50 = 672 nM T78709 CHO9C0 49864292 IC50 = 280 nM T78709 C8TB6G 49864336 Ki = 62 nM T78709 C5N8ML 49864359 Ki = 27.4 nM T78709 C15NIO 49864360 Ki = 102 nM T78709 C90MTG 49864602 IC50 = 3399 nM T78709 C5BCS4 49864722 IC50 = 95 nM T78709 CKZO79 49864723 IC50 = 3756 nM T78709 C74LZS 49864724 IC50 = 485 nM T78709 C2RY0J 50878551 Ki = 19 nM T78709 C1W6TV 50898777 Ki > 10000 nM T78709 CXMZ73 50898778 Ki > 10000 nM T78709 C67IRJ 50908804 Ki = 1.585 nM T78709 CLOB24 50908805 Ki = 1.259 nM T78709 CA89QH 50914389 Ki = 32.8 nM T78709 CX48AD 51002362 EC50 > 10000 nM T78709 C6LVM3 51003382 Ki = 3 nM T78709 CIW56N 51003383 Ki = 3 nM T78709 C8TA1J 51003550 IC50 = 1598 nM T78709 CQ1UJ7 51003551 IC50 = 1210 nM T78709 CGMI37 51003586 IC50 = 999 nM T78709 CE4KP1 51050257 Ki > 10000 nM T78709 C2HGK8 51122451 Ki = 30 nM T78709 CIWA18 52938727 Ki = 7.59 nM T78709 C6XY8V 52938728 Ki = 9.68 nM T78709 C9C0NB 52940734 Ki = 17.5 nM T78709 CLW3B0 52940951 Ki = 31.62 nM T78709 CWYS78 52941004 Ki = 5.012 nM T78709 CE0X9W 52941056 Ki = 7.943 nM T78709 C0UXM7 52941358 Ki = 2.09 nM T78709 CTM81E 52941423 Ki = 2.61 nM T78709 C40WVE 52941624 Ki = 2.512 nM T78709 CV7HZ6 52942047 Ki = 6.918 nM T78709 C5Y3VS 52942152 Ki = 15.85 nM T78709 CX9AF4 52942551 Ki = 0.3981 nM T78709 CE6R7D 52942615 Ki = 0.615 nM T78709 CR0G5U 52942644 Ki = 0.631 nM T78709 CX2E5H 52942854 Ki = 13.4 nM T78709 CU8WA5 52942916 Ki = 0.838 nM T78709 CO9J6M 52943356 Ki = 3.981 nM T78709 CLJ70C 52943589 EC50 = 32 nM T78709 CCF97B 52943811 Ki = 1 nM T78709 C2FG9O 52943861 Ki = 0.3981 nM T78709 C9G4CI 52943891 Ki = 1.259 nM T78709 C9RD4F 52944256 Ki = 35 nM T78709 CBU2Z6 52944379 Ki = 0.67 nM T78709 CRL3P0 52944615 Ki = 31.62 nM T78709 C4N6ET 52944674 Ki = 12.59 nM T78709 CCVP06 52944840 Ki = 3.162 nM T78709 C59ASG 52945060 Ki = 2.13 nM T78709 CDQ27E 52945156 Ki = 3.162 nM T78709 C7VQ5U 52945241 EC50 = 47 nM T78709 CHX9A2 52945310 Ki = 65.8 nM T78709 CPI9F4 52945803 Ki = 31.62 nM T78709 C4SH8M 52945840 Ki = 1.98 nM T78709 COM4R0 52946036 EC50 = 48 nM T78709 CJ49MX 52946290 Ki = 3.981 nM T78709 CRIV53 52946792 Ki = 1.08 nM T78709 C4S8JC 52946835 Ki = 0.803 nM T78709 CGZ1R7 52947088 Ki = 15.85 nM T78709 CS3OD1 52947342 Ki = 0.312 nM T78709 CCOQ59 52947343 Ki = 4.25 nM T78709 C6YB2T 52947380 Ki = 0.814 nM T78709 CK5ER0 52947414 Ki = 0.631 nM T78709 CNH57S 52947579 Ki = 15.85 nM T78709 CAVB03 52947615 Ki = 1 nM T78709 C1HRK4 52947622 Ki = 1 nM T78709 CS01XE 52947712 EC50 = 600 nM T78709 CD17LV 52948101 Ki = 1.44 nM T78709 CX04NC 52948119 Ki = 11.22 nM T78709 C7IR4Q 52948256 Ki = 0.517 nM T78709 CXR12O 52948486 EC50 = 18 nM T78709 CJ6OP5 52948620 Ki = 1.68 nM T78709 C4ZC1K 52948697 Ki = 0.631 nM T78709 C9YBJ3 52948823 Ki = 2.512 nM T78709 CLOB90 52949351 Ki = 3.61 nM T78709 CCQZ15 52949448 Ki = 15.14 nM T78709 C0RUM1 52949810 Ki = 2.34 nM T78709 CS6O4B 52949885 Ki = 3.22 nM T78709 CILY85 52950060 Ki = 0.786 nM T78709 CPVM58 52950169 Ki = 0.859 nM T78709 CT7A6Q 52952304 Ki = 50.12 nM T78709 CHC1S3 52952422 Ki = 3162.28 nM T78709 C4MZ1V 53237227 Ki = 1100 nM T78709 CBIL92 53237431 Ki = 2500 nM T78709 C7L6PJ 53237434 Ki = 2800 nM T78709 C9UX5B 53237437 Ki = 130 nM T78709 CMV78H 53237440 Ki = 39 nM T78709 CL73GJ 53237662 Ki = 240 nM T78709 CS02ZU 53237664 Ki = 2500 nM T78709 C5MLV8 53237666 Ki = 140 nM T78709 CLUD12 53237668 Ki = 100 nM T78709 C9P7KL 53237670 Ki = 59 nM T78709 C8T9OE 53237672 Ki = 14 nM T78709 COJM04 53237674 Ki = 160 nM T78709 C4TNP6 53237891 Ki = 68 nM T78709 C9RIJ7 53237893 Ki = 53 nM T78709 CBZX08 53237895 Ki = 68 nM T78709 C5ZT7N 53237897 Ki = 75 nM T78709 C4KRV8 53237899 Ki = 31 nM T78709 CNJ02E 53237901 Ki = 330 nM T78709 C0H6TR 53237903 Ki = 78 nM T78709 C8TDE6 53238121 Ki = 94 nM T78709 CN4R7I 53238123 Ki = 210 nM T78709 CIP64Q 53238125 Ki = 78 nM T78709 C70LGK 53238127 Ki = 420 nM T78709 C2WK6F 53238129 Ki = 2700 nM T78709 C6C0KM 53238131 Ki = 1400 nM T78709 CXN12U 53238133 Ki = 540 nM T78709 C9QXC8 53238134 Ki = 120 nM T78709 C9Z3FA 53238355 Ki = 310 nM T78709 C1Z8AH 53238357 Ki = 65 nM T78709 CMJ62D 53245590 Ki = 400 nM T78709 C4IV2J 53248158 Ki = 49 nM T78709 C03JEZ 53248159 Ki = 159 nM T78709 C2G0ZY 53248208 Ki = 37.9 nM T78709 C2UKM3 53248209 Ki = 1150 nM T78709 C8KW9J 53248210 Ki = 73 nM T78709 C87SLP 53248211 Ki = 501 nM T78709 CVD7E5 53248212 Ki = 101 nM T78709 CX6KG9 53248213 Ki = 223 nM T78709 C63MQD 53248256 Ki = 299 nM T78709 CG2O7F 53248257 Ki = 6000 nM T78709 CRK87G 53248258 Ki = 139 nM T78709 C73WQX 53248259 Ki = 2140 nM T78709 CKOV84 53248260 Ki = 1170 nM T78709 CGY45S 53248361 Ki = 1.11 nM T78709 CC9B3X 53248362 Ki = 1.11 nM T78709 CR4MN8 53248363 Ki = 0.87 nM T78709 CE9L8G 53248365 Ki = 0.64 nM T78709 C6KAR5 53248408 Ki = 1.95 nM T78709 CZG35A 53248409 Ki = 0.47 nM T78709 CGQJ07 53316788 Ki = 4 nM T78709 CZTW58 53317736 Ki = 22 nM T78709 CW70NZ 53318092 Ki = 30 nM T78709 C7PC1G 53318093 Ki = 8 nM T78709 CQ37BK 53318094 Ki = 19 nM T78709 C8RLQ9 53318095 Ki = 13 nM T78709 C5FRP2 53319428 Ki = 12 nM T78709 CY65NV 53319429 Ki = 6 nM T78709 C1MD0J 53319430 Ki = 16 nM T78709 C1E7BF 53319431 Ki = 90 nM T78709 C2OJW5 53319432 Ki = 1 nM T78709 CT0W3X 53319433 Ki = 203 nM T78709 C61DNP 53320009 IC50 = 672 nM T78709 C9ZDR5 53320010 IC50 = 333 nM T78709 CLQ85U 53322027 Ki = 8 nM T78709 C53HJK 53322028 Ki = 4 nM T78709 CQLK01 53322638 IC50 = 1226 nM T78709 CRUF31 53322954 Ki = 193 nM T78709 C2OB7G 53323389 Ki < 3 nM T78709 C4UBX5 53323390 Ki = 16 nM T78709 C1WU4E 53323391 Ki = 693 nM T78709 C32YWL 53324045 Ki = 481 nM T78709 CFJ1B0 53324709 Ki = 64 nM T78709 C35GJZ 53325137 Ki = 58 nM T78709 CRQF15 53325242 Ki = 1395 nM T78709 CZ69OW 53326010 Ki = 57 nM T78709 CZ1U9T 53326011 Ki = 14 nM T78709 C0UC1W 53326601 Ki = 7.5 nM T78709 C7MQZ6 53362652 Ki = 94 nM T78709 C4VW1I 53362653 Ki = 87 nM T78709 C24DBU 53362654 Ki = 89 nM T78709 CBF2P3 53362655 Ki = 96 nM T78709 C9MK6L 53362715 Ki = 124 nM T78709 C47KPJ 53362716 Ki = 90 nM T78709 C7PA6D 53362719 Ki = 276 nM T78709 CMB23T 53362720 Ki = 380 nM T78709 C7K0PH 53362779 Ki = 249 nM T78709 C8GC1B 53362840 Ki = 217 nM T78709 CU7W2I 53362841 Ki = 259 nM T78709 CH34LM 53362842 Ki = 137 nM T78709 CU4B6N 53370045 Ki = 489 nM T78709 CG24AT 53381002 Ki = 1354 nM T78709 C7WKR1 53387673 Ki > 10000 nM T78709 CFB1N5 53387674 Ki > 10000 nM T78709 CEIG81 53391632 Ki = 2540 nM T78709 CMOZ61 53475319 Ki = 708 nM T78709 C43VJF 54296648 Ki = 9.2 nM T78709 CEQ3M6 54579954 Ki = 2.15 nM T78709 C7WRB0 54579955 Ki = 1.68 nM T78709 C9VZ5P 54580443 Ki = 5 nM T78709 CQ4SI9 54580444 Ki = 9 nM T78709 C0R1QM 54581512 Ki = 851.14 nM T78709 C6PK2X 54582466 Ki = 15 nM T78709 CNW7S4 54582467 Ki = 7 nM T78709 C8V6BJ 54584468 Ki = 108 nM T78709 CY9QZ8 54584591 Ki = 0.6 nM T78709 CYX4S7 54585356 Ki = 11 nM T78709 CTQ08M 54586179 Ki = 3.5 nM T78709 CL5I1R 54753271 Ki = 1510 nM T78709 CG3UJ4 54758298 Ki = 6.7 nM T78709 COZ82F 55479093 Ki = 237 nM T78709 C8WHT5 56593934 Ki = 10000 nM T78709 CW89BT 56595402 Ki > 1000 nM T78709 C4C3XQ 56595529 Ki > 1000 nM T78709 CA54LD 56597090 Ki = 0.6 nM T78709 C6W1RA 56649648 Ki = 0.2 nM T78709 C2SW7J 56649649 Ki = 0.65 nM T78709 CQTR49 56649650 Ki = 0.86 nM T78709 CH37LU 56663451 IC50 > 10000 nM T78709 CR1OB6 56850389 EC50 = 16.3 nM T78709 CF63GQ 56850658 EC50 = 123 nM T78709 CJKO58 56852956 Ki = 40 nM T78709 CK7I9Z 56935084 Ki = 0.58 nM T78709 C20WGQ 56935085 Ki = 0.75 nM T78709 C17IZE 56935086 Ki = 0.74 nM T78709 CB0P9N 56944383 Ki = 110 nM T78709 C1ST9U 56944860 Ki = 4 nM T78709 CQKL90 56944861 Ki = 7 nM T78709 CS5J6Y 56944862 Ki = 10 nM T78709 CFLB40 56944863 Ki = 1.7 nM T78709 C53OTR 56944864 Ki = 6 nM T78709 C5T3RI 56944951 Ki = 5 nM T78709 CR6H7U 56944952 Ki = 12 nM T78709 C1Y2RP 56944953 Ki = 9 nM T78709 C1BH7I 56944954 Ki = 4 nM T78709 CTK9I8 56944955 Ki = 4 nM T78709 CCF1A5 56944956 Ki = 1 nM T78709 C2YVT8 56945042 Ki = 16 nM T78709 CNI2G3 56945043 Ki = 7.4 nM T78709 CCW38Z 56945164 Ki = 0.3236 nM T78709 CN6XE8 56945165 Ki = 0.5623 nM T78709 CPE6C7 56945166 Ki = 9.55 nM T78709 C4L7GW 56945167 Ki = 0.7943 nM T78709 CL68PZ 56946472 Ki = 1.995 nM T78709 CJ98DO 56946474 Ki = 0.8318 nM T78709 CB8J2F 56946573 Ki = 4.365 nM T78709 CCBY53 56946575 Ki = 10.47 nM T78709 CMO0U3 56946577 Ki = 3.467 nM T78709 CJZ3P4 56946579 Ki = 3.467 nM T78709 C1TC7Q 56963799 Ki > 10000 nM T78709 CUL4N1 56964693 Ki = 375 nM T78709 CQ5TP0 56964794 Ki = 19 nM T78709 CDGZ96 57326583 Ki = 266 nM T78709 C20ILW 57326584 Ki = 131 nM T78709 CD9I4N 57334553 IC50 = 11.8 nM T78709 C6H9UV 57345617 Ki = 102 nM T78709 CZU6L2 57345618 Ki = 73 nM T78709 CK9G8H 57345619 Ki = 91 nM T78709 C1US6F 57345626 Ki = 147.91 nM T78709 CD50GK 57345628 Ki = 10.47 nM T78709 C4FA1T 57345629 Ki = 14.79 nM T78709 C19DPJ 57381099 Ki = 711 nM T78709 CHD7U6 57381100 Ki = 10600 nM T78709 CL4Q2R 57381101 Ki = 776.5 nM T78709 C5ASK3 57381102 Ki = 1100 nM T78709 CZYV86 57381316 Ki = 221 nM T78709 C7U6SI 57381317 Ki = 2100 nM T78709 C0EW2L 57381318 Ki = 59000 nM T78709 C2F1UZ 57381319 Ki = 1400 nM T78709 CKIW81 57381320 Ki = 3200 nM T78709 CR9MZ4 57384073 Ki = 0.8 nM T78709 CATM39 57390694 Ki = 216 nM T78709 C6S0IE 57390695 Ki = 495 nM T78709 CCU1S2 57390881 Ki = 15 nM T78709 CV08WY 57391216 Ki = 93.1 nM T78709 CD75YK 57391306 Ki = 613 nM T78709 C07PMA 57391307 Ki = 80 nM T78709 CWT20M 57393083 Ki = 8.6 nM T78709 CDTG05 57393527 Ki = 22.91 nM T78709 CADH19 57394285 Ki = 168 nM T78709 C0WA3H 57394810 Ki = 454 nM T78709 CD4A3P 57396484 Ki = 23 nM T78709 C4EXS6 57396571 Ki = 154 nM T78709 C2ZWS1 57398007 Ki = 1.1 nM T78709 CR1Y7M 57398332 Ki > 10000 nM T78709 C3GW6L 57398351 Ki = 169 nM T78709 CO50ZB 57398352 Ki = 1080 nM T78709 CJ41PW 57399432 Ki = 263 nM T78709 CO3B4P 57399494 Ki = 415 nM T78709 C5GPJ0 57401515 Ki = 6.5 nM T78709 CG8MF3 57401516 Ki = 324 nM T78709 CZX05B 57401706 Ki = 6.2 nM T78709 CYN38R 57401819 Ki = 112 nM T78709 CO0XD2 57401820 Ki = 166 nM T78709 C8EFT7 57402251 Ki = 9.333 nM T78709 CL02EQ 57403172 Ki = 1.82 nM T78709 CX0B5M 57403525 Ki = 658 nM T78709 CWBG94 57403981 Ki = 274 nM T78709 CQB6F9 57456630 Ki = 85 nM T78709 C0M5PN 57873490 Ki > 1000 nM T78709 CH1BN8 57873491 Ki = 43 nM T78709 CI5UO1 57873492 Ki = 59 nM T78709 C2D9HA 57873499 Ki > 1000 nM T78709 C81MLX 57873504 Ki = 24 nM T78709 C7L9IE 57873508 Ki = 2 nM T78709 CZRL39 57873513 Ki > 1000 nM T78709 C98WTS 57873515 Ki = 2 nM T78709 C6BHT3 57873518 Ki = 94 nM T78709 CPX17D 57873520 Ki = 0.7 nM T78709 C54ROE 57873522 Ki = 26 nM T78709 CM7PI1 57873525 Ki = 9.9 nM T78709 CMUR21 57873527 Ki = 117 nM T78709 CO5Y9Q 57873531 Ki = 4 nM T78709 CZI37P 58760107 Ki = 10.91 nM T78709 CYSV60 60165411 Ki = 3.6 nM T78709 CB9GC6 60165412 Ki = 3.6 nM T78709 CI5PM3 60165413 Ki = 7.3 nM T78709 C2Q5VD 60165416 Ki = 90.5 nM T78709 C9JL3F 60165418 Ki = 6.6 nM T78709 C31PEN 60165535 Ki = 5.1 nM T78709 CP60YF 60165537 Ki = 111 nM T78709 CP1DR8 60165539 Ki > 10000 nM T78709 C85OTH 60165541 Ki = 85 nM T78709 CJO91V 60165543 Ki = 63 nM T78709 CJDC53 60165545 Ki = 214 nM T78709 C3K5JN 60165681 Ki = 28.3 nM T78709 C5RUP6 60167166 Ki = 312 nM T78709 CRH49P 60167309 Ki = 771 nM T78709 CX0NY3 60167310 Ki = 350 nM T78709 COHK72 60167451 Ki = 251.19 nM T78709 C30SVG 60167452 Ki = 102.33 nM T78709 CB4HT7 60195992 Ki = 63.2 nM T78709 C6VWY1 60196073 Ki = 31.4 nM T78709 C18AVJ 60196075 Ki = 14.9 nM T78709 CIN29U 60196077 Ki = 149 nM T78709 C5N3SG 60196080 Ki = 17.4 nM T78709 CI30FT 60204111 Ki = 10 nM T78709 CWSA08 60204112 Ki = 44 nM T78709 CLXS32 66561333 Ki = 226.8 nM T78709 CM24PO 66561413 Ki = 0.58 nM T78709 CN30YT 66800947 Ki = 1 nM T78709 CZ3MR6 66800959 Ki = 110 nM T78709 C92CMO 66800965 Ki = 3 nM T78709 C3K8DC 66801052 Ki = 21 nM T78709 C41VYW 66801295 Ki = 10 nM T78709 CR2N0J 66801344 Ki = 70 nM T78709 C3RX4C 66801425 Ki = 96 nM T78709 C7JD0I 66801429 Ki = 70 nM T78709 CN8OU1 66801430 Ki = 110 nM T78709 COR1H8 66801528 Ki = 36 nM T78709 C1F3YV 66801537 Ki = 18 nM T78709 C75WXP 66801561 Ki = 10 nM T78709 CC8JV6 66801624 Ki = 280 nM T78709 C3EI2F 66801625 Ki = 520 nM T78709 C0XG6B 66801701 Ki = 170 nM T78709 C42EBQ 66801837 Ki = 470 nM T78709 CW3AI2 66803474 Ki = 1.8 nM T78709 CPKH06 66803497 Ki = 11 nM T78709 CNJE57 66803500 Ki = 10 nM T78709 CN6FZ1 66803595 Ki = 6.1 nM T78709 C1LEH8 67268994 Ki > 10000 nM T78709 CD3U6K 68731121 Ki = 9720 nM T78709 C6IP8Q 69082816 Ki = 9040 nM T78709 CKM14W 69432471 Ki = 206 nM T78709 CP9V6A 69836292 Ki = 1995.26 nM T78709 CZ41VT 70683643 Ki = 125.8 nM T78709 C6EI2D 70684206 Ki = 730.02 nM T78709 CND4A2 70685780 Ki = 5.78 nM T78709 C6W9UK 70685781 Ki = 0.95 nM T78709 C4REJ6 70687910 Ki = 7.53 nM T78709 C4QNS1 70689942 Ki = 902.6 nM T78709 C0D7IM 70689943 Ki = 122.5 nM T78709 CY1BV3 70689944 Ki = 397.9 nM T78709 CBD3K8 70690497 Ki = 599.89 nM T78709 C8YMI5 70692100 Ki = 95.3 nM T78709 C9J3TO 70692655 Ki > 5000 nM T78709 CJQX48 70693375 Ki = 39.81 nM T78709 CIEG52 70694142 Ki = 159.8 nM T78709 CR7OD5 70694143 Ki = 4.73 nM T78709 C9HV4J 70694144 Ki = 1.39 nM T78709 CU4EK1 70694145 Ki = 2.26 nM T78709 C76JRL 70694146 Ki = 0.5 nM T78709 CET05I 70694683 Ki = 66 nM T78709 CTF76B 70694687 Ki > 1000 nM T78709 CST13M 70695474 Ki = 5.754 nM T78709 CQZ38N 70696271 Ki = 2264 nM T78709 CS7UT3 70697522 Ki = 569 nM T78709 CR5KY1 71061607 Ki = 877 nM T78709 C72XPZ 71061659 Ki = 1274 nM T78709 CKE2Y4 71061750 Ki = 614 nM T78709 CD1ET2 71061756 Ki = 918 nM T78709 C5KM2W 71061887 Ki = 239 nM T78709 C0D5SC 71062035 Ki = 35 nM T78709 CNQ65S 71062123 Ki = 80 nM T78709 CBF6Z8 71109804 Ki > 5000 nM T78709 C68NPQ 71109805 Ki = 208 nM T78709 CC43QK 71151588 Ki = 6.7 nM T78709 CJZ81X 71293954 Ki = 0.8 nM T78709 CZ35EN 71294092 Ki = 0.66 nM T78709 C6VL7X 71449080 Ki = 5.11 nM T78709 CKN5D4 71449120 Ki = 85.5 nM T78709 C91SZN 71449641 Ki = 290 nM T78709 C2GCN7 71449642 Ki = 65 nM T78709 CQN93U 71449643 Ki = 92 nM T78709 CEJ3B4 71449644 Ki = 10 nM T78709 C5SAJ1 71449645 Ki = 89 nM T78709 CG06AP 71449737 Ki = 2.48 nM T78709 C3XNC2 71450247 Ki = 8836 nM T78709 CDI84E 71450922 IC50 > 10000 nM T78709 CHT21G 71451454 Ki = 841 nM T78709 C2QZL4 71451455 Ki = 18 nM T78709 CXI5Q2 71451456 Ki = 456 nM T78709 CKJZ57 71451457 Ki = 21 nM T78709 C0F1HU 71451458 Ki = 5 nM T78709 CTZ24N 71451459 Ki = 49 nM T78709 C70JUP 71451460 Ki = 75 nM T78709 C9WLY7 71452692 Ki = 0.91 nM T78709 CUK2P5 71453252 Ki = 190 nM T78709 CKI58Z 71453278 Ki = 48 nM T78709 C1QM8D 71453279 Ki = 717 nM T78709 C6O4KT 71453280 Ki = 81 nM T78709 CL49VI 71453281 Ki = 31 nM T78709 CGXT64 71453282 Ki = 147 nM T78709 C7SQ0I 71453386 Ki = 14.01 nM T78709 CE0R9D 71454275 Ki = 5709 nM T78709 C0R2UV 71454458 Ki = 1.05 nM T78709 CGO13Q 71454997 Ki = 101 nM T78709 C0K1JV 71454998 Ki = 104 nM T78709 C3JF1D 71454999 Ki = 436 nM T78709 C2QZ1N 71455000 Ki = 313 nM T78709 C6FE5D 71455001 Ki = 230 nM T78709 C4L0JN 71455002 Ki = 22 nM T78709 CQSA61 71455082 Ki = 35.85 nM T78709 C8YH0J 71455083 Ki = 0.51 nM T78709 CAQF34 71455625 Ki = 4987 nM T78709 CD8O2C 71456208 Ki = 7.82 nM T78709 CWR40I 71456780 Ki = 283 nM T78709 CZUX67 71456781 Ki = 45 nM T78709 CZ17FC 71456782 Ki = 9 nM T78709 CKF09U 71456783 Ki = 22 nM T78709 CJKV72 71456784 Ki = 32 nM T78709 C82HSE 71456889 Ki = 1.89 nM T78709 C1PHO6 71456890 Ki = 16.29 nM T78709 C7MNB5 71457264 EC50 > 1000 nM T78709 CMJ1O9 71457409 Ki = 5629 nM T78709 C3GKR6 71458006 Ki = 4.45 nM T78709 CX06FZ 71458032 Ki = 24.55 nM T78709 CPO82B 71458050 Ki = 158.49 nM T78709 C84QJC 71458071 Ki = 510 nM T78709 C37EBC 71458647 Ki = 141 nM T78709 CM6OP1 71458648 Ki = 903 nM T78709 CRGE05 71458649 Ki = 270 nM T78709 CJN4S1 71458650 Ki = 28 nM T78709 CNT5J9 71458651 Ki = 23 nM T78709 C3NAM7 71458652 Ki = 10 nM T78709 CI6H3T 71458739 Ki = 1.61 nM T78709 CS83IF 71459269 Ki = 680 nM T78709 C3OR6K 71459910 Ki = 1.23 nM T78709 CG0WO9 71459954 Ki = 234 nM T78709 CT17XB 71460468 Ki = 30 nM T78709 CMOF94 71460561 Ki = 8.27 nM T78709 C63YLA 71461049 Ki > 10000 nM T78709 CJD96I 71461050 Ki > 10000 nM T78709 C6VL5X 71461632 Ki = 22.7 nM T78709 C0E9NL 71461634 Ki = 33.88 nM T78709 C7AX1Q 71462178 Ki = 45 nM T78709 C1CS0Z 71462179 Ki = 13 nM T78709 CHJ27Z 71462265 Ki = 36.19 nM T78709 CLP8D6 71462266 Ki = 8.36 nM T78709 C4P3JU 71462776 Ki > 10000 nM T78709 C3GUQ2 71462777 Ki > 10000 nM T78709 CD9G8B 71521478 Ki = 0.5495 nM T78709 CSV0G5 71521479 Ki = 0.309 nM T78709 CGN2M7 71521480 Ki = 0.3981 nM T78709 CT2ME3 71574204 Ki = 59 nM T78709 C3SXR5 71574206 Ki = 23 nM T78709 C2YRI9 71574208 Ki = 25 nM T78709 C62RWV 71574210 Ki = 14 nM T78709 CKC53S 71574212 Ki = 23 nM T78709 CNV42M 71574298 Ki = 88 nM T78709 C9PGQ1 71574300 Ki = 79 nM T78709 C2LXH5 71574302 Ki = 17 nM T78709 C2YPB8 71574304 Ki = 112 nM T78709 CK7GM0 71574306 Ki = 34 nM T78709 CI0GU8 71660496 IC50 > 48500 nM T78709 C0W2YA 71727193 Ki = 24 nM T78709 C79TLS 71727194 Ki = 15840 nM T78709 CFB10W 71727195 Ki = 1671 nM T78709 C6CIB5 71727196 Ki = 429 nM T78709 C7Z3JS 71727308 Ki = 117 nM T78709 CU5R1S 71758594 Ki = 243 nM T78709 C3ATN5 72197484 IC50 = 394.8 nM T78709 C20HSN 72197485 IC50 = 1252 nM T78709 CN8A5R 72197486 IC50 = 1057 nM T78709 CL3BF7 72197668 IC50 = 822.8 nM T78709 CWH6T3 72548703 IC50 = 0.43 nM T78709 C8Z0NM 72550642 Ki = 20 nM T78709 CL6W2Q 72550645 Ki = 11 nM T78709 C78LYM 72698087 Ki > 10000 nM T78709 C63HPK 72698088 Ki > 10000 nM T78709 C4AS0E 72699528 Ki = 1.3 nM T78709 CO20CN 72699532 Ki = 11 nM T78709 C8EVJ6 72699690 Ki = 3.9 nM T78709 CEAK86 72699692 Ki = 1.2 nM T78709 CIR7G1 72699716 EC50 = 590 nM T78709 CRMC07 72699718 Ki = 777.79 nM T78709 COH4F8 72699779 Ki = 15 nM T78709 C4X9AO 72699812 Ki = 997.7 nM T78709 C5K9JW 72699815 Ki = 553.1 nM T78709 CIDS43 72699817 EC50 = 850 nM T78709 C6J8GM 72699818 Ki = 175.32 nM T78709 CC8PL5 72699903 Ki = 285.33 nM T78709 C7YTK9 72699904 Ki = 654.64 nM T78709 C26STM 72700473 Ki = 0.69 nM T78709 CL96GC 72700475 Ki = 1.1 nM T78709 C45JKS 72700476 Ki = 5.6 nM T78709 C3TO8B 72700557 Ki = 1.7 nM T78709 CVA2X7 72700634 Ki = 2.1 nM T78709 C0KTL6 72734840 IC50 = 1200 nM T78709 CIO0W1 72734841 IC50 = 599 nM T78709 CTG91B 72734842 IC50 = 15 nM T78709 C49FUQ 72734843 IC50 = 16 nM T78709 C4E6PH 72734844 IC50 = 7200 nM T78709 CU9E5O 72734845 IC50 = 4500 nM T78709 CS48GA 72735019 IC50 = 5700 nM T78709 CB8CJ9 72735020 IC50 = 4900 nM T78709 C2WXK6 72735021 IC50 = 128 nM T78709 CC6Q5R 72771081 Ki < 100 nM T78709 C5L8NJ 72947314 Ki = 83.18 nM T78709 CE1JY2 72947315 Ki = 79.43 nM T78709 CC65OA 73213195 Ki = 371.54 nM T78709 CW83DK 73213196 Ki > 10000 nM T78709 C02FTM 73291731 Ki = 13.8 nM T78709 CCV91B 73346042 Ki = 0.1 nM T78709 CRG9J8 73346332 Ki > 10000 nM T78709 CM3IA6 73349341 EC50 = 45 nM T78709 C1MTL3 73350910 EC50 = 1195 nM T78709 CSCJ76 73350911 EC50 = 19 nM T78709 CD9Y0J 73350915 EC50 = 76 nM T78709 CL38VQ 73351112 Ki > 1000 nM T78709 CR0D1A 73356945 EC50 = 23 nM T78709 CVF5P0 73603034 IC50 = 4900 nM T78709 CUB97Z 74538690 Ki = 582 nM T78709 C2E7QW 75201901 Ki = 1200 nM T78709 C8IDL3 75306277 Ki = 39.81 nM T78709 CX17RZ 76280896 Ki = 203 nM T78709 C45OSP 76284193 Ki = 1055 nM T78709 C0CRJ1 76284452 Ki = 568 nM T78709 CS17IJ 76284453 Ki = 875 nM T78709 CH82JU 76284455 Ki = 272 nM T78709 CRO7Q9 76284721 Ki = 433 nM T78709 C4BIC2 76284724 Ki = 152 nM T78709 C0EKY7 76284725 Ki = 961 nM T78709 CS3HT5 76309671 Ki = 100 nM T78709 CXJG08 76314094 Ki = 387 nM T78709 CE5C2B 76319004 Ki = 25.7 nM T78709 C5F1XU 76321735 Ki = 700 nM T78709 C5TQ0X 76322648 Ki = 26.73 nM T78709 C94VNF 76324975 Ki = 537 nM T78709 CZ6P1E 76328545 Ki = 186 nM T78709 CGBE87 76335066 Ki = 90.2 nM T78709 CW3AK0 76335863 Ki = 743 nM T78709 C1UZ5J 76441180 Ki = 5.3 nM T78709 C28RIZ 76518514 Ki = 102 nM T78709 C8EWX5 85658088 Ki = 1805 nM T78709 C70ZVB 86221574 Ki = 5396 nM T78709 CJ9N5Q 86280005 Ki = 2.5 nM T78709 CJ92WR 86288399 Ki = 3.67 nM T78709 CMJA85 86288474 Ki = 1.1 nM T78709 C9S0XK 86288947 Ki = 121 nM T78709 CEPC94 86288948 Ki = 121 nM T78709 CJ9K3T 86290953 IC50 = 3800 nM T78709 CUA89I 86341962 Ki = 0.2 nM T78709 CWPH45 86341996 Ki = 1.4 nM T78709 CCR8X7 86342061 Ki = 12 nM T78709 CY2I8J 86342094 Ki = 5.2 nM T78709 CC47HJ 86342098 Ki = 5.3 nM T78709 CK03YC 86342156 Ki = 1.3 nM T78709 C5AQK2 86342192 Ki = 1.1 nM T78709 C9DZ2I 86342193 Ki = 0.52 nM T78709 CQP38R 86342194 Ki = 7.6 nM T78709 CE39OD 86342294 Ki = 1.1 nM T78709 C9T3LW 89638708 EC50 = 0.3 nM T78709 CHE2U4 90178632 Ki = 437 nM T78709 CD7R6P 90213677 Ki = 7.2 nM T78709 CWMU25 90644511 IC50 = 500 nM T78709 C37CYS 90654670 Ki = 122 nM T78709 C0IQ5R 90654671 Ki = 18 nM T78709 CVG2C1 90654672 Ki < 1 nM T78709 CU0ON1 90654673 Ki = 2 nM T78709 CJR3Y9 90654674 Ki = 122 nM T78709 CO1H4U 90654675 Ki = 107 nM T78709 CAY64Z 90654676 Ki = 12 nM T78709 CH0R8B 90654677 Ki = 77 nM T78709 CRFB56 90654678 Ki = 72 nM T78709 CPR21O 90654679 Ki = 236 nM T78709 C6YLV3 90654680 Ki = 499 nM T78709 CGUY51 90654681 Ki = 211 nM T78709 CK8X4O 90654682 Ki = 1914 nM T78709 CH8UQ9 90654683 Ki = 643 nM T78709 CTQ23Z 90654684 Ki = 16 nM T78709 C9Q2JW 90654685 Ki = 212 nM T78709 C98TJR 90654686 Ki = 377 nM T78709 CG3OI7 90654687 Ki = 230 nM T78709 CKTV83 90654688 Ki = 89 nM T78709 CVK85U 90654689 Ki = 47 nM T78709 CLG75D 90654690 Ki = 14 nM T78709 C7T9HW 90654691 Ki = 23 nM T78709 C92BZL 90654692 Ki = 313 nM T78709 C6CD9R 90654693 Ki = 214 nM T78709 C6H9NV 90654694 Ki = 44 nM T78709 CR74SD 90654695 Ki = 6307 nM T78709 C7VM4O 90654696 Ki = 52 nM T78709 CGFU53 90654697 Ki = 232 nM T78709 C7BEZ8 90654698 Ki = 141 nM T78709 CZ3IM2 90654699 Ki = 38 nM T78709 C8TMK5 90654700 Ki = 573 nM T78709 C7GK3C 90654701 Ki = 83 nM T78709 CN8BO1 90654702 Ki = 4 nM T78709 CHIW63 90654703 Ki = 2908 nM T78709 C1SAW2 90654704 Ki = 214 nM T78709 CJG31T 90654831 Ki = 5.5 nM T78709 CMU45O 90654832 Ki = 13.2 nM T78709 C14NPE 90654833 Ki = 135 nM T78709 C3C4BW 90654834 Ki = 124 nM T78709 C8QWR3 90654835 Ki = 23.3 nM T78709 C6ZR9L 90654837 Ki = 79 nM T78709 C0AC7R 90654839 Ki = 26 nM T78709 CKLG40 90654841 Ki = 45 nM T78709 C5JS8D 90654843 Ki = 76 nM T78709 C4VHZ6 90654845 Ki = 201 nM T78709 CG78PS 90654847 Ki = 235 nM T78709 CL39WP 90654849 Ki = 299 nM T78709 C0TVQ9 90654851 Ki = 305 nM T78709 C4I1CU 90654853 Ki = 88 nM T78709 CZ28YC 90654855 Ki = 301 nM T78709 CRO83N 90654857 Ki = 2178 nM T78709 CI91AM 90655807 Ki = 105 nM T78709 CY3L4T 90655808 Ki = 11.1 nM T78709 C2FG8Q 90655809 Ki = 2.62 nM T78709 C4R6CT 90655810 Ki = 14 nM T78709 CUQ8E6 90655811 Ki = 9.3 nM T78709 CU94HP 90655812 Ki = 7.55 nM T78709 CVY16X 90655813 Ki = 6.1 nM T78709 C12JSA 90655814 Ki = 33.5 nM T78709 CNB86Y 90655815 Ki = 42.5 nM T78709 C7NW4X 90655816 Ki = 221.4 nM T78709 CHG3S1 90655817 Ki = 31.6 nM T78709 C93XMI 90655818 Ki = 28.95 nM T78709 CANR17 90655819 Ki = 7.29 nM T78709 C58SPJ 90655820 Ki = 21 nM T78709 CB2ZL6 90655821 Ki = 8.06 nM T78709 CTZP78 90655822 Ki = 631 nM T78709 C23KCF 90655823 Ki = 425 nM T78709 CJSZ89 90655824 Ki = 496 nM T78709 CCOV98 90664359 Ki = 13340 nM T78709 C4MUI2 90664601 IC50 = 4.9 nM T78709 CXD5Q9 90664621 Ki = 4503 nM T78709 CKM05S 90664904 IC50 > 10000 nM T78709 CHT7D5 90664962 IC50 = 3.9 nM T78709 CACG19 90666899 Ki = 489.78 nM T78709 CODM50 90666903 Ki = 102.33 nM T78709 CSRU41 91242334 EC50 = 21.3 nM T78709 C0J5YH 91864602 Ki = 8.128 nM T78709 CRX16J 91884611 EC50 = 9.75 nM T78709 CDWS84 91937906 Ki < 1 nM T78709 CUQ6V0 92042918 Ki < 1000 nM T78709 CE0ZC6 101876962 Ki = 1174.9 nM T78709 C4DG3V 102364516 Ki > 1000 nM T78709 C4WDR8 109018769 Ki = 0.34 nM T78709 CF0XJ6 109018934 Ki = 938 nM T78709 CYB18Z 109027017 Ki = 272 nM T78709 CP6F4D 112815120 Ki = 305 nM T78709 CSH7K4 117949705 Ki = 118.7 nM T78709 C0M3CD 118051679 Ki = 13 nM T78709 CEMZ15 118464420 Ki = 320 nM T78709 CV2L6O 118464425 Ki = 116 nM T78709 CFNG86 118464427 Ki = 6764 nM T78709 CMSN80 118626035 Ki = 13 nM T78709 CT3AI0 118626042 Ki = 8 nM T78709 CKNJ72 118626045 Ki = 10 nM T78709 CGB42Y 118626088 Ki = 5 nM T78709 C0XJT5 118626089 Ki = 18 nM T78709 CIE4C7 118626101 Ki = 6 nM T78709 C1NYS5 118626120 Ki = 6 nM T78709 CPG04R 118626121 Ki = 13 nM T78709 C3S5LJ 118626129 Ki = 15 nM T78709 CY3F0N 118626140 Ki = 66 nM T78709 CE07IQ 118626142 EC50 = 11 nM T78709 C72OZY 118626161 Ki = 24 nM T78709 CY3E7S 118626169 Ki = 7 nM T78709 CHRB75 118626208 Ki = 6 nM T78709 C2Q4OP 118709739 Ki = 523 nM T78709 CZ68PL 118709740 Ki = 576 nM T78709 CSB25E 118709750 Ki = 13 nM T78709 CD4S9R 118709751 Ki = 8.2 nM T78709 CBP52O 118709752 Ki > 1000 nM T78709 CO72SF 118709753 Ki = 470 nM T78709 CJQR81 118709754 Ki = 491 nM T78709 CPW1D5 118709755 Ki > 1000 nM T78709 C1TMO7 118709756 Ki > 1000 nM T78709 CZDE01 118713090 Ki = 190 nM T78709 C1KR9C 118713091 Ki = 180 nM T78709 CI5U1R 118713092 Ki = 220 nM T78709 C4S7WD 118713093 Ki = 0.46 nM T78709 CB8Q2E 118713094 Ki = 0.835 nM T78709 CH9W0A 118713587 Ki = 913 nM T78709 CK43CN 118713588 Ki = 24.58 nM T78709 CL0TS7 118713589 Ki = 10.36 nM T78709 C4RD6F 118713590 Ki = 695.11 nM T78709 CIG13W 118713591 Ki = 83.33 nM T78709 CX5L1H 118713592 Ki = 6.13 nM T78709 CDWY84 118713593 Ki = 74.92 nM T78709 CO5S1I 118713594 Ki = 19.22 nM T78709 CI91US 118713595 Ki = 95.66 nM T78709 CW92LT 118713679 Ki = 11.86 nM T78709 C8P9YT 118713680 Ki = 7.13 nM T78709 CZ1K5R 118713681 Ki = 3.96 nM T78709 CH7ZE8 118713682 Ki = 0.91 nM T78709 CKX78H 118713683 Ki = 1.3 nM T78709 C5LSA7 118713684 Ki = 0.43 nM T78709 CPAI54 118713685 Ki = 29.78 nM T78709 C6U2LR 118713686 Ki = 0.27 nM T78709 CYA6E4 118713687 Ki = 0.19 nM T78709 CZ9UL2 118713688 Ki = 0.21 nM T78709 CUV5Y0 118715454 EC50 > 30000 nM T78709 CI7NQ9 118716698 Ki = 9.333 nM T78709 CGO9W4 118716699 Ki = 46.77 nM T78709 CVDI36 118716700 Ki = 14.45 nM T78709 C94AFL 118716701 Ki = 117.49 nM T78709 CTX92K 118716702 Ki = 81.28 nM T78709 CG02WP 118716703 Ki = 158.49 nM T78709 CTNL85 118716704 Ki = 15.85 nM T78709 CM1Y8W 118716705 Ki = 8.913 nM T78709 C42MOT 118716706 Ki = 58.88 nM T78709 C78ARU 118716707 Ki = 50.12 nM T78709 CO5TG3 118716708 Ki = 42.66 nM T78709 CNF78L 118716709 Ki = 20.42 nM T78709 C9CB1Q 118716710 Ki = 36.31 nM T78709 C3F6EQ 118716711 Ki = 64.57 nM T78709 C0L6YO 118716712 Ki = 323.59 nM T78709 CX2AC4 118716713 Ki = 52.48 nM T78709 CL1EU8 118716714 Ki = 26.92 nM T78709 C0V7GJ 118716715 Ki = 37.15 nM T78709 CRBI65 118716716 Ki = 69.18 nM T78709 C70IPZ 118716717 Ki = 24.55 nM T78709 CBI30N 118716718 Ki = 43.65 nM T78709 C7UBN8 118716719 Ki = 60.26 nM T78709 CV8HA2 118716720 Ki = 144.54 nM T78709 C30ZJB 118716721 Ki = 33.11 nM T78709 C58MND 118716722 Ki = 79.43 nM T78709 CO6T4G 118716723 Ki = 87.1 nM T78709 C8RVX4 118717455 Ki = 616.6 nM T78709 C5IM1N 118717456 Ki = 3467 nM T78709 CBCU90 118717457 Ki = 891 nM T78709 CN4LJ2 118717458 Ki = 1096 nM T78709 CZ35PU 118717459 Ki = 1380 nM T78709 C9BP7A 118717460 Ki = 1258.93 nM T78709 CFCM61 118717461 Ki = 2818 nM T78709 C8C6ZW 118717462 Ki = 602.56 nM T78709 CG0O3Q 118719795 Ki = 6 nM T78709 CUHT71 118719796 Ki = 5.8 nM T78709 CR0FM7 118719797 Ki = 7.4 nM T78709 CPX2Y1 118719798 Ki = 1.3 nM T78709 C0KH8S 118719799 Ki = 153 nM T78709 CWO13F 118719807 Ki = 9.4 nM T78709 CUH0A6 118719810 Ki = 3.9 nM T78709 CES97Y 118722639 Ki = 15 nM T78709 CM3P7R 118722912 Ki = 67 nM T78709 CP3QC2 118722913 Ki = 11 nM T78709 C1PG3C 118722914 Ki = 73 nM T78709 CR6E5D 118722915 Ki > 1000 nM T78709 CGA86P 118728506 Ki = 39.6 nM T78709 C9PGE7 118728507 Ki = 37.4 nM T78709 CR4GE1 118728510 Ki = 15.2 nM T78709 C14LZH 118728511 Ki = 363 nM T78709 C14RAC 118728513 Ki = 114 nM T78709 CQK04P 118728514 Ki = 53.9 nM T78709 CK9CG4 118728521 Ki = 28.9 nM T78709 C1N9JU 118728522 Ki = 268 nM T78709 C1UZ8G 118728523 Ki = 6.28 nM T78709 CPCE84 118728524 Ki = 51.5 nM T78709 CBN06J 118728525 Ki = 1.04 nM T78709 CF3QE0 118728526 Ki = 16.1 nM T78709 CJG4Q1 118728527 Ki = 211 nM T78709 C4NFW1 118728528 Ki = 3.23 nM T78709 CO8LF9 118728529 Ki = 26.4 nM T78709 CCN7R8 118728530 Ki = 1.03 nM T78709 C5O2NU 118729733 Ki = 3842 nM T78709 CTE58Z 118730369 Ki = 500 nM T78709 CB3Y2W 118731347 Ki = 16 nM T78709 CWZF06 118731348 Ki = 53 nM T78709 CA3O1H 118731349 Ki = 34 nM T78709 CU8P4W 118731350 Ki = 20 nM T78709 C8GKX6 118731351 Ki = 66 nM T78709 C2J4VC 118731352 Ki = 26 nM T78709 CF7NH5 118731353 Ki = 61 nM T78709 CQ8F6C 118731354 Ki = 1 nM T78709 CR9J0O 118731355 Ki = 17 nM T78709 CU12XM 118731356 Ki = 35 nM T78709 C4CEV7 118731357 Ki = 18 nM T78709 CU6T2D 118731358 Ki = 9 nM T78709 C95WKJ 118731359 Ki = 35 nM T78709 C20QAO 118731360 Ki = 16 nM T78709 CT6J8V 118731361 Ki = 14 nM T78709 C7QVJ4 118731362 Ki = 47 nM T78709 CA2X3O 118731363 Ki = 36 nM T78709 C4DV8I 118731364 Ki = 19 nM T78709 CHVY82 118731365 Ki = 40 nM T78709 CM5FG1 118731366 Ki = 16 nM T78709 C7W3EY 122178698 Ki = 506 nM T78709 CF8P1H 122178699 Ki = 153 nM T78709 C48MFR 122178700 Ki = 179 nM T78709 CZ72QS 122178701 Ki = 273 nM T78709 C4VY8A 122178702 Ki = 845 nM T78709 C2KF4Z 122178703 Ki = 563 nM T78709 CX6MJ2 122178704 Ki = 244 nM T78709 CA53KF 122178705 Ki = 117 nM T78709 C8XD3F 122178706 Ki = 152 nM T78709 CTRC59 122178707 Ki = 224 nM T78709 C5QV8D 122178708 Ki = 163 nM T78709 C84UED 122178709 Ki = 361 nM T78709 CV96JK 122178710 Ki = 92 nM T78709 CM89KS 122178711 Ki = 102 nM T78709 CXL5V3 122183764 Ki = 9 nM T78709 CK3VT8 122183765 Ki = 21 nM T78709 C12TRH 122183771 Ki = 84 nM T78709 C06GQO 122183778 Ki = 68 nM T78709 C3VDY7 122197403 Ki = 13 nM T78709 C1MFJ3 122197404 Ki = 13 nM T78709 CBHT01 122377930 Ki = 356 nM T78709 CLW53P 122483274 Ki = 22 nM T78709 CO63ET 122483280 Ki = 122 nM T78709 C4QM2E 124247485 Ki = 1866 nM T78709 CM57GR 126720252 Ki = 5650 nM T78709 CLWM12 126720394 Ki = 1354 nM T78709 C8Q1JB 126720403 Ki = 5934 nM T78709 C1U3SZ 126720425 Ki = 2277 nM T78709 C5G8FD 126720440 Ki = 2790 nM T78709 CD50YM 127024949 Ki = 23 nM T78709 C4GF2D 127024950 Ki = 46 nM T78709 CJ76IB 127024951 Ki = 206 nM T78709 CIHZ54 127025242 Ki = 142 nM T78709 CCY7P3 127025243 Ki = 98 nM T78709 CNJ4Z1 127025244 Ki = 99 nM T78709 CTBN56 127026052 Ki = 79.43 nM T78709 C26NMB 127026071 Ki = 1847 nM T78709 C1YD7M 127026119 Ki = 463 nM T78709 CUO7Y8 127026120 Ki = 197 nM T78709 CDU21O 127026131 Ki = 51 nM T78709 C9HDP8 127026132 Ki = 431 nM T78709 CTYP30 127026133 Ki = 254 nM T78709 C19BOM 127026141 Ki = 947 nM T78709 CZFB49 127026142 Ki = 199 nM T78709 C2FT3B 127026143 Ki = 148 nM T78709 CP4J5H 127026144 Ki = 591 nM T78709 C6BIU4 127026145 Ki = 190 nM T78709 C1FA2U 127026146 Ki = 718 nM T78709 CE43NR 127026147 Ki = 502 nM T78709 C1TV0X 127026296 Ki > 1000 nM T78709 CDAP16 127026434 Ki = 6147 nM T78709 C2XO3L 127026443 Ki = 4570 nM T78709 C80QHX 127026444 Ki = 556 nM T78709 CBF64M 127026450 Ki = 123 nM T78709 CO1FB4 127026451 Ki = 170 nM T78709 CC13RA 127026452 Ki = 74 nM T78709 CBE56W 127026514 Ki = 549 nM T78709 C0SZI4 127026515 Ki = 148 nM T78709 CS1WZ7 127026552 Ki > 1000 nM T78709 C67GCU 127026601 Ki = 7.586 nM T78709 C68ZHE 127026602 Ki = 7.244 nM T78709 C94PCX 127026603 Ki = 50.12 nM T78709 C03TAB 127026604 Ki = 125.89 nM T78709 C3MEP4 127026605 Ki = 416.87 nM T78709 C7P0YF 127026609 Ki > 1000 nM T78709 C1SV6Z 127026610 Ki > 1000 nM T78709 C3V1WR 127026611 Ki > 1000 nM T78709 CX6EI2 127026750 Ki = 545 nM T78709 CEG15O 127026751 Ki = 373 nM T78709 C1J4QY 127026752 Ki = 28 nM T78709 C0WB2U 127026753 Ki = 45 nM T78709 C9AWR7 127026894 Ki > 1000 nM T78709 CQC3H0 127026895 Ki > 1000 nM T78709 CSA2O0 127026896 Ki > 1000 nM T78709 CIG2V3 127027195 Ki > 1000 nM T78709 CC9O6J 127027196 Ki > 1000 nM T78709 C4R5SE 127027197 Ki > 1000 nM T78709 C0UOJ6 127027386 Ki = 371 nM T78709 C9IH1A 127027387 Ki = 407 nM T78709 C0TC7E 127027388 Ki = 536 nM T78709 CZ4W6I 127027389 Ki = 393 nM T78709 C4YR7A 127027390 Ki = 260 nM T78709 C3FA0I 127027391 Ki = 2667 nM T78709 CSHA70 127027488 Ki > 1000 nM T78709 CQJZ73 127027489 Ki > 1000 nM T78709 CZT84N 127027491 Ki > 1000 nM T78709 CNBO79 127027492 Ki > 1000 nM T78709 CJB98N 127027493 Ki > 1000 nM T78709 C3VO6E 127027494 Ki > 1000 nM T78709 CMT35D 127027495 Ki > 1000 nM T78709 CO21RS 127027496 Ki > 1000 nM T78709 CC71UE 127027715 Ki = 1068 nM T78709 CY2TW9 127028152 Ki = 2733 nM T78709 CAZJ04 127028153 Ki = 2969 nM T78709 CR48GO 127028154 Ki = 1646 nM T78709 C8MC1I 127028408 Ki = 750 nM T78709 CD8H7W 127028471 Ki = 397 nM T78709 C4EAY5 127028472 Ki = 98 nM T78709 CUS8R9 127028473 Ki = 319 nM T78709 CA10BY 127028634 Ki = 745 nM T78709 C7JD9S 127028726 Ki = 162.18 nM T78709 C31GSQ 127028730 Ki = 549.54 nM T78709 CZ26YR 127028797 Ki = 59 nM T78709 CI2R1N 127028798 Ki = 1304 nM T78709 CS8GJ5 127028799 Ki = 6862 nM T78709 CU0WQ3 127029375 Ki = 5298 nM T78709 CS1GX5 127029649 Ki = 9167 nM T78709 C9N3BE 127029650 Ki = 821 nM T78709 CQFS48 127029651 Ki = 1004 nM T78709 C7F3YE 127029652 Ki = 5570 nM T78709 CZ61LK 127034966 IC50 > 5011.87 nM T78709 CA0SN5 127034967 IC50 = 1995.26 nM T78709 CQ0ZT9 127035062 Ki = 821 nM T78709 CU49VE 127036186 Ki = 31.62 nM T78709 CG06BD 127036932 Ki = 58.88 nM T78709 CVW71O 127036953 Ki = 10 nM T78709 C7N5DF 127037679 Ki = 208 nM T78709 CD13VY 127037680 Ki = 455 nM T78709 CTE43C 127037681 Ki = 616 nM T78709 C0LGK6 127037682 Ki = 103 nM T78709 C2XBE8 127037921 Ki = 17770 nM T78709 CX0CN4 127037922 Ki = 342 nM T78709 CXR71M 127038002 Ki = 2.455 nM T78709 CDAE15 127038033 Ki = 232 nM T78709 CFA6Q8 127038034 Ki = 74 nM T78709 CERL85 127038035 Ki = 279 nM T78709 C8TC9G 127038281 Ki = 159 nM T78709 CPK2Z7 127038282 Ki = 5555 nM T78709 CL5N3P 127038713 Ki = 40.74 nM T78709 CYJ2D5 127039593 Ki = 214 nM T78709 CQED51 127039753 Ki = 159 nM T78709 CL4E2K 127039754 Ki = 368 nM T78709 CES26L 127039755 Ki = 234 nM T78709 CQ36LP 127039756 Ki = 183 nM T78709 C89SOL 127040060 Ki = 3.802 nM T78709 CQ3L8Z 127040156 Ki = 3.02 nM T78709 C7KA2C 127040443 Ki = 278 nM T78709 CKBZ01 127040444 Ki = 249 nM T78709 CFAB12 127040760 Ki = 178 nM T78709 CWQ47G 127040761 Ki = 373 nM T78709 C8D4AV 127040908 Ki = 180 nM T78709 CE12AY 127041106 Ki = 321 nM T78709 C71LGS 127041107 Ki = 74 nM T78709 C6RI9V 127041108 Ki = 102 nM T78709 C15BGV 127041244 Ki = 140 nM T78709 CU0J4S 127041258 Ki = 190 nM T78709 C20MZH 127041259 Ki = 346 nM T78709 CP16CZ 127041260 Ki = 2346 nM T78709 CZT53S 127041261 Ki = 4511 nM T78709 C0FJP2 127041563 Ki = 9054 nM T78709 CUC3F9 127041564 Ki = 9626 nM T78709 COG9D2 127041874 Ki = 62 nM T78709 CS4WH1 127042184 Ki = 30 nM T78709 C13AIN 127042185 Ki = 80 nM T78709 CR59TP 127042539 Ki = 158 nM T78709 C54IZC 127042540 Ki = 249 nM T78709 C8G1HF 127042841 Ki = 14030 nM T78709 C0V5YU 127048532 EC50 = 361 nM T78709 CHW0L2 127048533 EC50 = 120 nM T78709 C9QR6V 127048539 EC50 = 6 nM T78709 CU6K4P 127048540 EC50 = 8.2 nM T78709 CC7BU0 127049059 Ki = 380.19 nM T78709 C42FHY 127049060 Ki = 376 nM T78709 CF2QY9 127049061 Ki = 1162.5 nM T78709 CN2F1W 127049163 EC50 = 12 nM T78709 C1TI6J 127049515 EC50 = 7.2 nM T78709 CT16PL 127049516 EC50 = 122 nM T78709 C4QKS3 127049517 EC50 = 26 nM T78709 C03BLH 127049522 EC50 = 309 nM T78709 C2IX7Q 127049847 EC50 = 34.4 nM T78709 CRK8W3 127049848 EC50 = 97.2 nM T78709 C85PIF 127049849 EC50 = 137 nM T78709 CO2V5Z 127049850 EC50 > 10000 nM T78709 C27MWC 127049861 EC50 = 122 nM T78709 CZS1L6 127049862 EC50 = 13 nM T78709 CZD91J 127049863 EC50 = 13 nM T78709 C1S6EN 127049864 EC50 = 4.3 nM T78709 C2H0BQ 127049865 EC50 = 2.7 nM T78709 CUK1S9 127049866 EC50 = 5.1 nM T78709 CX53AC 127050632 Ki = 102 nM T78709 CP9UT4 127050764 EC50 > 100 nM T78709 C9T2VY 127050765 EC50 = 24 nM T78709 CIOZ65 127051038 EC50 = 26 nM T78709 C7XK3G 127051039 EC50 = 101 nM T78709 CR4TV6 127051040 EC50 = 464 nM T78709 CCTO35 127051041 EC50 = 74 nM T78709 CA2SJ6 127051340 EC50 = 301 nM T78709 CTL0S1 127051516 Ki = 194.98 nM T78709 CTL8J1 127051843 Ki = 295 nM T78709 CF6V9Q 127051844 Ki = 38 nM T78709 C8TNB1 127051845 Ki = 23 nM T78709 CT9O7G 127051863 Ki = 3153 nM T78709 C5ONG1 127051864 Ki = 251.19 nM T78709 CRF85X 127052458 Ki = 33.5 nM T78709 CCY71I 127052465 Ki = 533 nM T78709 C2E9VX 127052467 Ki = 1689 nM T78709 CPO4C3 127052468 Ki = 190.55 nM T78709 CSQ2N8 127052486 Ki = 611 nM T78709 CLU7C1 127052757 Ki = 141 nM T78709 C95KYT 127052758 Ki = 244 nM T78709 CYNR02 127052759 Ki = 217 nM T78709 C1JAS7 127052779 Ki = 33.88 nM T78709 C7MQK8 127053042 Ki = 40.74 nM T78709 C3WIA6 129103318 IC50 = 587.8 nM T78709 CBX2V6 129186527 EC50 > 10000 nM T78709 CV2K7I 129186528 EC50 = 24.22 nM T78709 CD9C1F 129186530 EC50 > 10000 nM T78709 C2F5YE 129186531 EC50 > 10000 nM T78709 C6GC0F 129186534 EC50 = 7.2 nM T78709 CTP0O3 129186549 EC50 = 34.1 nM T78709 C8KM6N 129186554 EC50 = 4.57 nM T78709 C7FR6U 129186558 EC50 = 899 nM T78709 CEZT92 129186564 EC50 = 7.09 nM T78709 C1CV2Y 129840786 Ki = 1.5 nM T78709 CJ5S2O 129840806 Ki = 809 nM T78709 C9K8MH 129840818 Ki = 6.7 nM T78709 C36AFR 129840841 Ki = 4.8 nM T78709 CUD71X 129840856 Ki = 33 nM T78709 CV4D2F 129840894 Ki = 250 nM T78709 C40HCZ 129840904 Ki = 8 nM T78709 CY7DS0 129840906 Ki = 1.7 nM T78709 CJX83W 129840907 Ki = 3500 nM T78709 C4PU0E 129840972 Ki = 1 nM T78709 C6K4NX 129840994 Ki = 60 nM T78709 C6Y7FB 129841007 Ki = 15 nM T78709 CKA0L7 129841015 Ki = 250 nM T78709 CK1G0Y 129841036 Ki = 0.7 nM T78709 CGUW90 129841059 Ki = 389 nM T78709 CV8SI7 129841063 Ki = 7 nM T78709 C10VDB 130431277 Ki = 70.3 nM T78709 CI1NF8 130431279 Ki = 3560 nM T78709 CS8O4E 130431287 Ki = 560 nM T78709 C85MOW 130431289 Ki = 910 nM T78709 C2OH7B 130431291 Ki = 2660 nM T78709 CEQ43Y 130431295 Ki = 9500 nM T78709 CK64GU 130431296 Ki = 117 nM T78709 CYW0X2 130431314 Ki = 248 nM T78709 CDN26V 130431316 Ki = 880 nM T78709 CL64UW 130431317 Ki = 27.6 nM T78709 C8HE2O 130431318 Ki > 7600 nM T78709 CZ6S4T 130431319 Ki = 131 nM T78709 C8ZHI7 130431325 Ki = 26 nM T78709 CF5SW8 130431328 Ki = 4980 nM T78709 CN9RZ3 130431329 Ki = 2800 nM T78709 CN70MW 130431337 Ki = 59 nM T78709 C4GF1U 130431342 Ki = 2410 nM T78709 C2WI5R 130431351 Ki = 2330 nM T78709 C50GOC 130442480 Ki = 6900 nM T78709 CM04RF 130442572 Ki = 2500 nM T78709 C1RI8Q 132060720 Ki = 2019 nM T78709 CY8B9L 132060743 Ki = 2609 nM T78709 C4VNA6 132060746 Ki = 2135 nM T78709 CGHO19 132060770 Ki = 335 nM T78709 CT81OY 132060776 Ki = 1201 nM T78709 CFXL21 132060812 Ki = 733 nM T78709 C4LJ2Y 132503215 Ki = 45 nM T78709 CM8B1L 132525569 Ki = 1501 nM T78709 CU5L0K 132525570 Ki = 637 nM T78709 CA10SQ 132547275 Ki = 17.4 nM T78709 C6E1GN 132547276 Ki = 6.96 nM T78709 C6VTW3 132547277 Ki = 8.21 nM T78709 CI70OP 132547278 Ki = 25.9 nM T78709 C3Q1LA 132547279 Ki = 2.99 nM T78709 CAVB41 132584404 Ki > 10000 nM T78709 CS0MB3 132938109 Ki = 1329 nM T78709 C8O2EP 134130246 Ki = 95 nM T78709 C8M9FH 134130379 Ki = 111 nM T78709 CA4GX3 134130447 Ki = 33.5 nM T78709 C7ZDA2 134130462 Ki = 18.6 nM T78709 CWL50Q 134130594 Ki = 167 nM T78709 C8TG2O 134130846 Ki = 100 nM T78709 CHP3J4 134131015 Ki = 90.3 nM T78709 CQ4IF8 134131147 Ki = 17.8 nM T78709 C6N5FS 134131151 Ki = 772 nM T78709 CH4XB2 134131159 Ki = 1032 nM T78709 CR32SP 134131265 Ki = 52.1 nM T78709 C0JKL5 134131283 Ki = 24.7 nM T78709 C3Z6SV 134131949 Ki = 4500 nM T78709 C0RQC6 134131976 Ki = 2870 nM T78709 C6D1HC 134132279 Ki > 1000 nM T78709 CQX4U3 134133064 Ki = 338.84 nM T78709 C2V8BH 134133118 Ki = 1.96 nM T78709 CCPI30 134133464 Ki = 2.3 nM T78709 CTS3J4 134133483 Ki = 105 nM T78709 C0J2ML 134133604 Ki = 15.49 nM T78709 CM4XE8 134133829 Ki = 2.239 nM T78709 C6QAF1 134133900 IC50 < 10 nM T78709 CM0TS6 134133967 Ki = 29 nM T78709 CC1DO8 134134456 Ki = 771 nM T78709 CR4F6X 134135492 Ki = 1.5 nM T78709 CM34TY 134135507 Ki = 3 nM T78709 C2Q3JY 134135516 Ki = 595 nM T78709 CJG3U0 134136134 Ki = 149 nM T78709 C3P9IJ 134136137 Ki = 9.4 nM T78709 CLA4R3 134136207 Ki = 2.27 nM T78709 CGX03A 134136246 Ki = 1096.48 nM T78709 C7L2SN 134136382 Ki = 6.04 nM T78709 CKH7W6 134137025 Ki = 5.012 nM T78709 C08ZBY 134137332 Ki = 1836 nM T78709 CD41CW 134137432 Ki = 2.9 nM T78709 CXF52V 134137560 Ki = 103 nM T78709 CN4LI8 134137732 Ki = 134 nM T78709 C5A6XO 134138438 Ki = 3.02 nM T78709 C90XZH 134138881 Ki = 15 nM T78709 CTP83K 134139510 Ki = 1.1 nM T78709 C7X6TJ 134139808 Ki = 5.4 nM T78709 CRC2V0 134139826 Ki = 2630 nM T78709 C8TC3Z 134140440 Ki = 2.12 nM T78709 CHK39T 134141166 Ki = 126 nM T78709 CLW86T 134141354 Ki = 1698.24 nM T78709 CXC80B 134142146 Ki = 1.3 nM T78709 C6PSI9 134142907 Ki = 3842 nM T78709 C46ZTY 134143085 Ki = 1.549 nM T78709 CVJ70S 134143778 Ki = 0.92 nM T78709 CR5L4K 134144303 Ki = 213.8 nM T78709 C80TGJ 134144864 Ki = 163 nM T78709 CWQG03 134145252 Ki = 0.81 nM T78709 CK37OV 134145259 Ki = 1.12 nM T78709 CK5RU9 134145903 Ki = 66 nM T78709 CLUV50 134145912 Ki = 1.4 nM T78709 C8AZ1F 134146083 Ki = 33 nM T78709 C8RI0E 134146106 Ki = 0.72 nM T78709 C2E0ID 134146185 Ki = 802 nM T78709 CC9P2T 134146194 Ki = 11 nM T78709 CV0QZ5 134147124 Ki = 365 nM T78709 C92WVK 134147870 Ki = 12.3 nM T78709 C41XSD 134147935 Ki = 6631 nM T78709 CL9RW7 134148069 Ki = 1.04 nM T78709 CBU81N 134149168 Ki > 10000 nM T78709 CEU53H 134149777 Ki = 0.9333 nM T78709 CA50EU 134150000 Ki = 29.3 nM T78709 CHK9J1 134150839 Ki = 1.56 nM T78709 CE6LN3 134151118 Ki = 74 nM T78709 CLU34D 134151427 Ki = 48.3 nM T78709 C2JN8Y 134151729 Ki = 202 nM T78709 CK23XB 134151891 Ki = 2.1 nM T78709 C76BZW 134151980 Ki = 160 nM T78709 CB14UF 134152029 Ki = 4 nM T78709 CIV4H5 134152583 Ki = 6064 nM T78709 CI0G7H 134153418 Ki = 39 nM T78709 CDWP64 134153527 Ki = 22.91 nM T78709 CB6M5Y 134153538 Ki = 41.69 nM T78709 CX4W7F 134153716 Ki = 109 nM T78709 C79TEI 134154068 Ki = 14.45 nM T78709 C9DQ4Y 134154208 Ki = 1.4 nM T78709 CMJ1U3 134154387 Ki = 138 nM T78709 CD80HF 134154490 Ki = 5 nM T78709 C4VGJ5 134154679 Ki = 9.9 nM T78709 C5SK4P 134154831 Ki = 0.36 nM T78709 CU6C4G 134154943 Ki = 5.3 nM T78709 C6QAY2 134155116 Ki = 18.62 nM T78709 C79QLN 134155460 Ki = 64.57 nM T78709 CIUZ94 134155476 Ki = 80 nM T78709 C90QNV 134155645 Ki = 101 nM T78709 CT5E7V 134155933 Ki = 2 nM T78709 CVR87Q 134156222 Ki = 122 nM T78709 CAB4K6 134156305 Ki = 147 nM T78709 C50XNE 134156520 Ki = 86 nM T78709 CUHE07 134157171 Ki = 160 nM T78709 C6S0VM 134157330 Ki = 3.02 nM T78709 CL6DN0 134157769 Ki = 152 nM T78709 C1GY2T 135156251 EC50 > 10000 nM T78709 C6N8GM 135367405 Ki > 10000 nM T78709 C6LU0C 135367816 Ki > 10000 nM T78709 CD2TH9 135367820 Ki > 10000 nM T78709 C5AMD9 135367857 Ki > 10000 nM T78709 CGBW93 135410312 Ki = 40.74 nM T78709 CVE08Y 135458392 Ki = 389 nM T78709 CP7HN4 135458393 Ki = 85 nM T78709 CS8XJ6 135458394 Ki = 246 nM T78709 C9B7XA 135458410 Ki = 124 nM T78709 CFV9A3 135458427 Ki = 240 nM T78709 CKX4N8 135458428 Ki = 53 nM T78709 C9ZCL5 135458672 Ki = 15560 nM T78709 C7DF4S 135464159 Ki = 323.59 nM T78709 CQDP70 135469307 Ki = 63 nM T78709 C7AGR0 135474338 Ki > 10000 nM T78709 CP9XN7 135500023 Ki = 11748.98 nM T78709 C34FXW 135501716 Ki = 2753 nM T78709 C6I9RK 135516645 Ki = 977.24 nM T78709 CQI23C 135516796 Ki = 1584.89 nM T78709 C3FV9I 135527031 Ki = 4168.69 nM T78709 CJF0P1 135600051 IC50 = 6.2 nM T78709 CD6L8Q 135895192 Ki = 1148 nM T78709 CA1M8B 135966709 Ki = 669 nM T78709 C6A8WK 136002690 IC50 = 46.6 nM T78709 C19GLK 136116062 Ki = 87 nM T78709 CA3JC8 136118613 Ki = 3445 nM T78709 CQ2GP6 136118614 Ki = 7361 nM T78709 C6R4IC 136118615 Ki = 7269 nM T78709 CS0JL5 136118616 Ki = 4608 nM T78709 C8RH6M 136118617 Ki = 2624 nM T78709 CHWC38 136118619 Ki > 10000 nM T78709 C5UDW3 136118620 Ki = 315 nM T78709 C8I6UN 136118621 Ki = 1812 nM T78709 C0W1TM 136118658 Ki = 6927 nM T78709 C40LYH 136118659 Ki = 2513 nM T78709 CZ7C3Y 136118660 Ki > 10000 nM T78709 C42FCS 136118661 Ki > 10000 nM T78709 CB12QP 136152964 Ki = 56 nM T78709 CFX06E 136152966 Ki = 348 nM T78709 C37YXA 136152971 Ki = 75 nM T78709 CY0C1X 136152972 Ki = 612 nM T78709 CSNE17 136179514 Ki = 478.63 nM T78709 CT0ZC8 136179515 Ki = 58.88 nM T78709 CX53NC 136180316 Ki = 36.6 nM T78709 CZ7WT9 136180317 Ki = 2.96 nM T78709 CQP2Y6 136180318 Ki = 75.3 nM T78709 CQT9H5 136180319 Ki = 43.5 nM T78709 CLPU18 136180320 Ki = 7.33 nM T78709 C0LO6Q 136180321 Ki = 116 nM T78709 C25RED 137631359 Ki = 0.5623 nM T78709 C9EIP8 137631570 EC50 = 30.8 nM T78709 CHM36P 137631892 Ki = 257 nM T78709 CVT4G8 137632024 Ki > 1000 nM T78709 CN1I7A 137634153 Ki > 20000 nM T78709 CC51JN 137635185 Ki > 10000 nM T78709 CNR82A 137635294 EC50 = 1300 nM T78709 C6DH9X 137635433 EC50 = 300 nM T78709 C0K3AP 137635725 EC50 > 10000 nM T78709 C94VXJ 137635884 Ki = 66 nM T78709 CFM92C 137636384 Ki > 10000 nM T78709 CF7KG5 137637817 Ki = 724 nM T78709 CDX39B 137637994 Ki = 370 nM T78709 C19JKQ 137638321 Ki = 1.122 nM T78709 CA03VC 137639125 Ki = 0.631 nM T78709 C1EK3W 137640451 Ki = 587 nM T78709 C3U5NF 137640522 EC50 = 680 nM T78709 CWQ80N 137640967 EC50 = 10.2 nM T78709 C3LYX9 137641832 Ki > 10000 nM T78709 C4I6QS 137641944 EC50 > 10000 nM T78709 C5WS6Q 137642134 Ki = 975 nM T78709 CU1O2P 137642386 Ki = 0.8913 nM T78709 CMJU75 137643395 EC50 = 28.6 nM T78709 CWUM83 137644521 Ki > 10000 nM T78709 CDA80E 137644790 Ki = 324 nM T78709 CHT42S 137645295 EC50 > 10000 nM T78709 CPCY48 137645406 Ki = 931 nM T78709 CZ8CU6 137645501 Ki = 40 nM T78709 CCP38D 137645926 Ki = 740 nM T78709 CVX74E 137646045 Ki = 5967 nM T78709 C96EAP 137646245 Ki = 0.6918 nM T78709 CPI68E 137646281 Ki = 0.22 nM T78709 C8PV0N 137646568 EC50 = 770 nM T78709 CO5U9A 137647674 EC50 = 1100 nM T78709 CMXI62 137649997 Ki = 749 nM T78709 CB4HG5 137650482 EC50 = 16.9 nM T78709 CWQF69 137650550 EC50 = 76.2 nM T78709 C52IRM 137650705 Ki = 54 nM T78709 CKG08R 137650961 Ki = 609 nM T78709 C47TWK 137651544 EC50 = 607 nM T78709 CW2L7Z 137651819 Ki = 0.7943 nM T78709 CU4S1W 137651887 Ki = 5 nM T78709 CVK26R 137652044 Ki = 543 nM T78709 CHFK13 137652210 Ki > 10000 nM T78709 C51CGJ 137652310 Ki = 759 nM T78709 C04XYN 137653567 EC50 = 10.5 nM T78709 C2E3FV 137653850 Ki = 32 nM T78709 C6N0DT 137654586 EC50 > 10000 nM T78709 CX82HS 137654666 Ki = 27 nM T78709 C0SKV1 137654850 Ki > 10000 nM T78709 C4VG0U 137655411 Ki = 29 nM T78709 CVEN03 137656381 EC50 = 69.7 nM T78709 CO3L7F 137656918 Ki > 10000 nM T78709 CEJ9L8 137657949 EC50 = 10.2 nM T78709 C3LHT5 137658253 EC50 = 32.9 nM T78709 C8G0HO 137658832 EC50 = 26.2 nM T78709 CFQ7C9 137659145 EC50 = 488 nM T78709 CLQX32 137659728 EC50 > 10000 nM T78709 CF9RZ5 137660385 EC50 = 450 nM T78709 CX4D7Y 137660741 Ki = 30 nM T78709 C9HPG8 137661516 IC50 = 600 nM T78709 C0R6XM 138691314 Ki = 1047 nM T78709 CU3Y7W 138691316 Ki = 1230 nM T78709 CH2W4P 138691317 Ki > 10000 nM T78709 CHSC40 138691321 Ki = 676 nM T78709 C18UZA 138691329 Ki = 9120 nM T78709 C1XWV0 138691338 Ki = 661 nM T78709 C6LE1A 138691362 Ki = 2138 nM T78709 CN9R4A 138691364 Ki = 123 nM T78709 C8H2KR 138691366 Ki = 2344 nM T78709 CJ43GI 139187858 Ki = 850 nM T78709 C47QCK 139187859 Ki = 3 nM T78709 C2Z9CD 139488518 Ki = 5623 nM T78709 CJK95T 139488527 Ki = 933 nM T78709 CZ6H9M 139488539 Ki = 316 nM T78709 CAF2H8 139488606 Ki = 589 nM T78709 C54CIL 139488740 Ki = 1738 nM T78709 CH7Y5D 141312275 Ki = 195 nM T78709 C4EU2S 141745651 Ki = 1.6 nM T78709 CCO6R0 141745657 Ki = 1.6 nM T78709 CO5DR9 145949220 Ki = 219 nM T78709 CWAF96 145949371 Ki = 85 nM T78709 CHG2W6 145950605 Ki = 305 nM T78709 COU57L 145950881 Ki = 140 nM T78709 CD4M6B 145951915 Ki = 18290 nM T78709 C5D1KR 145952639 EC50 = 1.2 nM T78709 C78AUI 145952711 Ki = 99 nM T78709 C8F3PN 145952866 EC50 > 10000 nM T78709 CA2J5S 145954503 Ki = 330400 nM T78709 C0JO8B 145954831 Ki = 421 nM T78709 CLJW61 145955880 Ki = 613 nM T78709 CHI1V8 145956064 Ki = 197 nM T78709 CSER68 145956892 Ki = 109 nM T78709 CLVI07 145957637 Ki = 18430 nM T78709 C91IDE 145958490 Ki = 341 nM T78709 C8VS7K 145959257 Ki = 2249 nM T78709 CSIZ31 145959706 Ki = 585 nM T78709 CD59BL 145960493 EC50 = 62.43 nM T78709 CXU82Q 145960544 EC50 = 93.37 nM T78709 CG8ZX0 145960719 EC50 < 0.14 nM T78709 CMO17A 145960744 Ki = 1.3 nM T78709 CQR07X 145960843 EC50 = 0.36 nM T78709 CDCS74 145960879 EC50 = 1563.21 nM T78709 CAJ7P6 145961144 Ki = 1 nM T78709 C59KNW 145961441 Ki = 2.2 nM T78709 CNF26K 145961458 EC50 = 34.98 nM T78709 CI4H8B 145961535 Ki = 92 nM T78709 C8PTZ7 145961730 Ki = 1 nM T78709 CP2M6G 145961773 EC50 = 0.58 nM T78709 CAE03F 145961788 EC50 = 28.8 nM T78709 CQ4RA7 145961842 Ki = 1.6 nM T78709 CBK15Q 145961968 EC50 = 0.35 nM T78709 C2TAU8 145962091 EC50 = 52 nM T78709 C1YE4Q 145962266 Ki = 1.5 nM T78709 CD6P4H 145962474 EC50 = 0.6 nM T78709 C8YS0D 145962581 EC50 = 0.75 nM T78709 C71HNB 145962633 Ki = 303 nM T78709 C7TM1V 145962678 EC50 = 146.01 nM T78709 C9G5YC 145962760 Ki = 253 nM T78709 C2A3DR 145962768 EC50 < 0.14 nM T78709 C56BKQ 145962801 Ki = 38 nM T78709 CVM9G4 145962946 Ki = 11 nM T78709 CFA09Q 145962985 Ki = 556 nM T78709 CO7P1B 145963059 Ki = 190 nM T78709 C4GS7B 145963079 EC50 = 0.72 nM T78709 CG94HV 145963146 EC50 = 1.55 nM T78709 C9B0SZ 145963169 Ki = 28 nM T78709 C2ZSA4 145963224 Ki = 1.6 nM T78709 CDTR93 145963270 Ki = 0.8 nM T78709 C4Y1PK 145963314 Ki = 100 nM T78709 CVM9W0 145963420 EC50 = 567 nM T78709 CHZ5I6 145963710 EC50 = 14.93 nM T78709 CNA8I5 145963810 Ki = 2 nM T78709 C7KC3T 145963830 IC50 > 10000 nM T78709 C5VWM7 145963860 Ki = 1169 nM T78709 CCK5G1 145963863 Ki = 1961 nM T78709 CEN94V 145963961 EC50 = 2.2 nM T78709 C3I6YP 145963975 EC50 > 100000 nM T78709 CV7YW9 145964086 Ki = 962 nM T78709 CE32PV 145964143 Ki = 5.4 nM T78709 CHDN35 145964150 IC50 > 10000 nM T78709 CR2B9G 145964154 Ki = 2058 nM T78709 C1KH2E 145964159 IC50 > 10000 nM T78709 C1B8QW 145964299 EC50 = 9 nM T78709 C7YKQ4 145964390 Ki = 8966 nM T78709 C95NZO 145964427 Ki = 32 nM T78709 C2P5NK 145964621 Ki = 1266 nM T78709 C0N8KC 145964622 EC50 = 28.1 nM T78709 CK0T1M 145964694 Ki = 742 nM T78709 C6T4RY 145964846 Ki = 20 nM T78709 C24NSP 145964857 Ki = 0.9 nM T78709 CE9K3L 145964944 Ki = 0.84 nM T78709 C7MBS0 145964982 EC50 > 100000 nM T78709 C7JS9I 145965041 EC50 = 117 nM T78709 C9D8IB 145965203 Ki = 2 nM T78709 C5DL3N 145965355 Ki = 14 nM T78709 C1MIR9 145965401 Ki = 496 nM T78709 CV07EO 145965433 EC50 > 100000 nM T78709 C9KXP6 145965474 Ki = 1350 nM T78709 CLP94W 145965668 Ki = 1096 nM T78709 C8TF9G 145965840 Ki = 13790 nM T78709 C53EFW 145966154 Ki = 388 nM T78709 CB05QA 145966199 Ki = 1322 nM T78709 CLM10C 145966333 EC50 = 1.2 nM T78709 C1T4DN 145966418 Ki = 2687 nM T78709 CRS7V6 145966748 Ki = 50 nM T78709 C5L4WF 145967359 EC50 = 17.6 nM T78709 CV03XA 145967457 Ki = 1951 nM T78709 CL58XS 145967572 Ki = 9.4 nM T78709 C58WSL 145967904 Ki = 272 nM T78709 C76SHX 145968149 Ki = 2.41 nM T78709 C3DZ7P 145968324 Ki = 42.8 nM T78709 C3D0LR 145968390 Ki = 11.3 nM T78709 CT09GI 145968506 Ki = 19.3 nM T78709 C9S8QE 145968791 Ki = 57.8 nM T78709 CB1FD8 145968810 Ki = 110 nM T78709 CM0Z9G 145968895 Ki = 2.25 nM T78709 CM6HG9 145968927 EC50 = 16.5 nM T78709 C2A0FO 145969167 EC50 > 100000 nM T78709 CVU49S 145969204 Ki = 19 nM T78709 CQ8EM6 145969402 Ki = 3755 nM T78709 CI5R8W 145969406 Ki = 0.5 nM T78709 CERC65 145969459 Ki = 69.9 nM T78709 CD3Z4I 145969495 Ki = 546 nM T78709 C48XNG 145969667 Ki = 15 nM T78709 CNZY06 145969934 Ki = 19 nM T78709 C3FNX8 145969978 Ki = 16 nM T78709 CRZN24 145970238 Ki = 251 nM T78709 CT2LQ4 145970743 Ki = 8.8 nM T78709 CQC6Y1 145970782 Ki = 1 nM T78709 C6FBU7 145970863 Ki = 43.1 nM T78709 C61MSO 145970938 Ki = 326 nM T78709 CF74MR 145971390 Ki = 1428 nM T78709 C1T7GL 145971527 Ki = 6100 nM T78709 CRC9T0 145971556 EC50 = 0.9 nM T78709 C8A2XG 145971561 Ki = 4054 nM T78709 CN64ZR 145971588 Ki = 770 nM T78709 CB43OV 145971604 Ki = 3.5 nM T78709 CQJ5O8 145971635 IC50 > 10000 nM T78709 C56RAO 145972025 Ki = 14900 nM T78709 C7BVC1 145972374 IC50 > 10000 nM T78709 CR06QO 145972382 EC50 > 100000 nM T78709 CWRM23 145972513 EC50 = 12.8 nM T78709 CJHI43 145972875 Ki = 1792 nM T78709 C1QY4E 145973003 Ki = 0.6 nM T78709 CS7WG8 145973438 Ki = 3198 nM T78709 C8KYV6 145973487 Ki = 2669 nM T78709 C0H1JO 145973539 Ki = 3168 nM T78709 CL74IP 145973853 Ki = 190 nM T78709 CT51VH 145974031 Ki = 0.9 nM T78709 CR0CX6 145974087 Ki = 184 nM T78709 C6AGN3 145974143 EC50 = 176 nM T78709 C8KZ5T 145974165 Ki = 6.3 nM T78709 C05IVJ 145974184 Ki = 8687 nM T78709 CW6EX3 145974189 Ki = 2081 nM T78709 C9L7EM 145974368 Ki = 2.5 nM T78709 CDOJ39 145974939 EC50 = 0.7 nM T78709 C3WG0J 145975106 Ki = 1630 nM T78709 CR83MU 145975214 EC50 = 23.6 nM T78709 C6PH4F 145975226 IC50 > 10000 nM T78709 CN8U3P 145975289 Ki = 1411 nM T78709 CJF4Z0 145975393 EC50 > 100000 nM T78709 CZ39GQ 145975595 EC50 > 100000 nM T78709 CSVR94 145975713 Ki = 4067 nM T78709 COY2P3 145975720 Ki = 14160 nM T78709 CL7EX5 145975776 Ki = 552 nM T78709 C1BI8E 145975778 Ki = 2368 nM T78709 C7R2MD 145975905 Ki = 6005 nM T78709 C71CYU 145975946 IC50 > 10000 nM T78709 C0V4AL 145975992 Ki = 52010 nM T78709 C2TN8W 145976085 IC50 > 10000 nM T78709 C8XFM7 145976120 Ki = 146 nM T78709 CF5B0W 145976158 Ki = 2211 nM T78709 CB2R6J 145976187 Ki = 1.5 nM T78709 C8BJI2 145976292 Ki = 1839 nM T78709 C90NFP 145976326 Ki = 1.48 nM T78709 CCDU50 145976348 EC50 = 42.3 nM T78709 CZ5XK2 145976408 Ki = 2891 nM T78709 C14OJW 145976618 Ki = 297 nM T78709 C0LRB2 145976686 Ki = 2677 nM T78709 C34XME 145976696 Ki = 5 nM T78709 CTCM92 145976698 Ki = 2349 nM T78709 CIZ69S 145976722 Ki = 462 nM T78709 C9FR7N 145976732 EC50 = 11.3 nM T78709 CNCS36 145976746 Ki = 3.7 nM T78709 CT7WO5 145976787 Ki = 4358 nM T78709 CI8AN3 145976890 Ki = 696 nM T78709 C81CSM 145976946 Ki = 1545 nM T78709 C8NW7Y 145977256 Ki = 3949 nM T78709 CHS96B 145977297 Ki = 2.4 nM T78709 C8DP4I 145977442 Ki = 11 nM T78709 C4L8EZ 145977467 Ki = 619 nM T78709 CC1DZ5 145977555 Ki = 2077 nM T78709 C0Y6QO 145977799 IC50 > 10000 nM T78709 CP8C6M 145978146 Ki = 506 nM T78709 C72SMR 145978208 EC50 = 6.2 nM T78709 C6HQI0 145978420 Ki = 509 nM T78709 C8VL3Y 145978472 Ki = 48240 nM T78709 C82NXP 145978482 Ki = 1456 nM T78709 C1Q2BR 145978965 EC50 = 17.4 nM T78709 C20XQJ 145979626 Ki = 6216 nM T78709 C2PK6X 145980101 Ki = 0.3 nM T78709 C87MSW 145980271 Ki = 1094 nM T78709 CW2CO4 145980458 Ki = 19 nM T78709 CD92WV 145980513 Ki = 1304 nM T78709 C8I7QL 145980875 Ki = 901 nM T78709 C6H7SC 145981004 Ki = 0.4 nM T78709 CC2UQ5 145981118 Ki = 186 nM T78709 C4AF0G 145981310 EC50 > 100000 nM T78709 C67AIW 145981408 EC50 = 2.4 nM T78709 CPK34X 145981875 Ki = 8.1 nM T78709 C7LBY5 145982138 Ki = 4 nM T78709 COY79P 145982165 Ki = 326 nM T78709 CO7WP6 145982353 EC50 = 10.5 nM T78709 CEK60A 145982506 Ki = 14 nM T78709 CI59TX 145983018 Ki = 23 nM T78709 CYC58R 145983059 Ki = 9 nM T78709 C4F5OT 145983128 Ki = 5 nM T78709 C5ZG9M 145983139 Ki = 179 nM T78709 CV2GU9 145983144 Ki = 146 nM T78709 C4PKM2 145983390 Ki = 50 nM T78709 C9LR8C 145983405 Ki = 18 nM T78709 CIAF74 145983468 Ki = 54 nM T78709 CE7MF4 145983751 Ki = 24 nM T78709 CDQ4U7 145983760 Ki = 12 nM T78709 CYW9B2 145983794 Ki = 12 nM T78709 C1DW4U 145983928 EC50 = 3.6 nM T78709 C8I1WG 145983961 Ki = 14 nM T78709 CP5H4D 145984065 Ki = 147 nM T78709 C58DHN 145984151 EC50 = 13.3 nM T78709 CJ35DM 145984299 Ki = 37 nM T78709 CU7E4M 145984511 Ki = 56 nM T78709 C6JUY0 145984737 Ki = 37 nM T78709 CID02G 145984807 Ki = 27 nM T78709 CP9D3A 145984902 Ki = 0.3 nM T78709 CM5X3V 145985050 Ki = 111 nM T78709 CG10LK 145985224 Ki = 48 nM T78709 CFJ9B3 145985233 Ki = 147 nM T78709 C5AOI6 145985289 Ki = 8 nM T78709 CW30NA 145985505 Ki = 86 nM T78709 C7ZRP1 145985527 Ki = 91 nM T78709 C2XY8Q 145985533 Ki = 25 nM T78709 C7NI4X 145985585 Ki = 96 nM T78709 C9LJ5T 145985692 Ki = 16 nM T78709 C7QIX0 145985718 Ki = 28 nM T78709 C6V5QS 145985823 Ki = 120 nM T78709 C07GKD 145985958 Ki = 36 nM T78709 CCM18E 145986031 Ki = 15 nM T78709 CR0XQ3 145986138 Ki = 16 nM T78709 CXC79K 145986552 EC50 = 47.9 nM T78709 COT25D 145986575 Ki = 468 nM T78709 CT37DW 145986720 Ki = 15150 nM T78709 CNJH37 145986752 Ki = 10000 nM T78709 C3VN5O 145987559 Ki = 5211 nM T78709 CZ5O8R 145987659 EC50 = 107 nM T78709 CI0PA9 145987771 Ki = 28 nM T78709 COS58J 145987942 EC50 = 10.6 nM T78709 C6MHU2 145988006 EC50 = 3.1 nM T78709 C9ZBE8 145988017 Ki = 3 nM T78709 CHOB70 145988038 EC50 = 1.6 nM T78709 CO4LK7 145988180 Ki = 12 nM T78709 CIS9P2 145988193 Ki = 62 nM T78709 C86XQR 145988313 Ki = 603 nM T78709 C9W1QA 145988497 EC50 = 8.8 nM T78709 CUGO10 145988693 Ki = 1262 nM T78709 C9D2OG 145988738 Ki = 129 nM T78709 C4C0YP 145988913 Ki = 21470 nM T78709 CDY48U 145989143 Ki = 0.53 nM T78709 CVC14L 145989181 EC50 = 91.3 nM T78709 CR2EV8 145989183 EC50 = 11.6 nM T78709 C39CSX 145989329 Ki = 154 nM T78709 CMJL94 145989451 EC50 = 6.1 nM T78709 CB6OP0 145989720 Ki = 8.76 nM T78709 C3GPR9 145990093 Ki = 377500 nM T78709 C41SBL 145990126 EC50 = 1.7 nM T78709 C2Q5UK 145990353 Ki = 128 nM T78709 CK5IA4 145990443 Ki = 6 nM T78709 CT7AB8 145990459 Ki = 5577 nM T78709 CE9PT1 145990482 EC50 = 3.3 nM T78709 C4GV8Q 145990586 Ki = 71 nM T78709 CKWF21 145990750 Ki = 1210 nM T78709 CMJ46R 145990794 EC50 = 6.9 nM T78709 CVBR36 145991084 Ki = 5.6 nM T78709 C5TNP0 145991127 EC50 = 1.1 nM T78709 CW14AE 145991244 EC50 > 100000 nM T78709 C7RJ4E 145991363 Ki = 11 nM T78709 CU6E1Z 145991746 EC50 = 13.8 nM T78709 C9TK6G 145991864 Ki = 15 nM T78709 CI1EQ3 145991900 Ki = 159 nM T78709 C9WME0 145992265 Ki = 0.4 nM T78709 CB8CM6 145992305 Ki = 1155 nM T78709 C5DVK4 145992403 Ki = 308 nM T78709 CCP2U1 145992489 Ki = 1363 nM T78709 CELG57 145992523 EC50 = 5.8 nM T78709 CLPU06 145992567 Ki = 413200 nM T78709 CB64KH 145992860 EC50 = 3.6 nM T78709 CBI94R 145992877 Ki = 13 nM T78709 C9PS8N 145993117 EC50 = 1.24 nM T78709 CT63XO 145993172 EC50 = 0.9 nM T78709 CI19KS 145993474 Ki = 25 nM T78709 C0Z6YX 145993493 EC50 = 7.7 nM T78709 C17HSV 145993577 EC50 = 1.2 nM T78709 C0TL8E 145993714 Ki = 1225 nM T78709 CX1N0L 145993740 Ki = 450 nM T78709 CO1BX3 145994087 Ki = 161 nM T78709 CS1LF2 145994186 Ki = 1.2 nM T78709 CC2G1V 146025727 Ki = 3700 nM T78709 C5ZOJ3 146680920 Ki = 5009 nM T78709 CG97ER 146709966 Ki = 2511.89 nM T78709 CF5B2L 147653864 Ki = 1000 nM T78709 C5PNX8 148302367 Ki = 1995.26 nM T78709 C9T0PS 153061504 Ki = 316.23 nM T78709 C1FA0K 153287541 Ki = 199.53 nM T78709 CEQ69Z 153287542 Ki = 199.53 nM T78709 C6P3SR 153287553 Ki > 10000 nM T78709 CW31CT 153287566 Ki = 199.53 nM T78709 CV9G7Z 153287572 Ki = 1995.26 nM T78709 CO85KL 153287574 Ki = 74 nM T78709 CZ1K4D 155510674 Ki = 4 nM T78709 CLX3D8 155510732 EC50 = 1180 nM T78709 CC3KP7 155510927 Ki > 10000 nM T78709 CM4RB0 155511262 Ki = 64 nM T78709 C0K7OA 155511383 EC50 > 100000 nM T78709 C9KX6O 155511928 Ki = 197 nM T78709 CZ7HP4 155512406 Ki = 993 nM T78709 C4OL0A 155512409 Ki = 5.15 nM T78709 C2H6LN 155512422 Ki = 52 nM T78709 CXF90M 155512487 Ki = 1010 nM T78709 C7N0VH 155512508 Ki > 1000 nM T78709 C1WG0H 155512850 EC50 = 100 nM T78709 CO68LC 155512944 Ki = 2344 nM T78709 C4Q5SY 155512981 Ki = 140 nM T78709 C90FST 155513438 Ki = 399 nM T78709 C36RDV 155513614 Ki = 327 nM T78709 C6DP0E 155513883 Ki = 218 nM T78709 C7W1OH 155513940 Ki = 1.549 nM T78709 C7FI9W 155514217 Ki = 84 nM T78709 CRP43D 155514341 IC50 > 1000 nM T78709 C95QOT 155514378 Ki = 2944 nM T78709 CK9YN0 155514430 Ki = 2260 nM T78709 CI4DT8 155514575 Ki = 126 nM T78709 CJUI87 155514774 Ki = 23 nM T78709 CM5A8F 155514858 Ki = 130 nM T78709 CQ84DA 155514889 Ki = 64 nM T78709 C21QLC 155515074 Ki = 63 nM T78709 CV8F7A 155515301 Ki = 12.02 nM T78709 C4X2RG 155515318 Ki = 431 nM T78709 C3NB0D 155515324 Ki > 1000000 nM T78709 C0Q8PR 155515407 Ki = 688 nM T78709 CWO56B 155515415 Ki > 10000 nM T78709 CU0PY6 155515687 Ki = 3.84 nM T78709 C2TN5D 155515890 Ki = 32 nM T78709 CW6O5J 155515898 Ki = 47 nM T78709 C7KT0D 155515919 Ki > 10000 nM T78709 C13LOV 155515942 Ki = 1872 nM T78709 CUM2N4 155515982 Ki = 17 nM T78709 C7OF4C 155516118 Ki = 6204 nM T78709 CG5M1O 155516282 Ki = 291 nM T78709 CG53LH 155516399 Ki = 40.4 nM T78709 C6X9UC 155516902 Ki = 76 nM T78709 CT4U8D 155517137 Ki = 28.18 nM T78709 CU8TC0 155517162 Ki = 12 nM T78709 CEA9D5 155517238 Ki = 157 nM T78709 CW0B5K 155518159 Ki > 10000 nM T78709 C87RWX 155518489 Ki = 431 nM T78709 CYB12O 155518974 Ki = 3569 nM T78709 CHVF41 155519045 Ki = 808 nM T78709 CCEZ93 155519102 Ki = 4540 nM T78709 CQD2J7 155519393 Ki = 1052 nM T78709 C2SXT1 155519515 Ki = 132 nM T78709 C0KLD8 155519559 Ki = 5036 nM T78709 CAV5Y1 155519565 Ki = 269.15 nM T78709 C07BTO 155519598 Ki = 54 nM T78709 CUSA24 155519891 Ki = 1000 nM T78709 C5FL7R 155520499 Ki = 482 nM T78709 C8OC3W 155520552 Ki = 149 nM T78709 CO1B0G 155520918 Ki = 233 nM T78709 CTV2F6 155521010 Ki > 1000 nM T78709 C17QKW 155521049 Ki = 134 nM T78709 CW0AM2 155521520 EC50 = 54400 nM T78709 CG2F9X 155521599 Ki = 261 nM T78709 CL07FB 155521817 Ki = 213.8 nM T78709 CWQ1D2 155521828 Ki = 378 nM T78709 CL20TG 155522125 EC50 > 100000 nM T78709 C98RDQ 155522218 Ki = 22 nM T78709 CAFT73 155522329 Ki = 68.7 nM T78709 CP6H1D 155522562 Ki = 46 nM T78709 CUQ61M 155522867 Ki = 21.2 nM T78709 CXEB36 155523275 Ki = 9.55 nM T78709 CD9QU6 155523519 Ki = 9 nM T78709 C2Y9CW 155523745 Ki = 220 nM T78709 C4NOD0 155524193 Ki = 1720 nM T78709 C5KYB4 155524228 Ki = 3.2 nM T78709 C7F2ZG 155524366 Ki = 240 nM T78709 CK4B0R 155524491 Ki = 8 nM T78709 CRF5T8 155524643 EC50 > 100000 nM T78709 CYZ60F 155524736 Ki = 70.79 nM T78709 CUO93F 155524808 Ki = 19 nM T78709 C65UZD 155524956 Ki = 106 nM T78709 CZQ5M2 155525523 Ki = 155 nM T78709 CR3DZ7 155525571 Ki = 203 nM T78709 CD5BI1 155525649 Ki = 5.248 nM T78709 C6MZJ9 155525703 Ki = 12 nM T78709 C81OCJ 155526014 Ki = 81.8 nM T78709 CZ81JA 155526026 Ki = 26 nM T78709 C68VNI 155526159 EC50 = 1600 nM T78709 CF7B3L 155526557 Ki = 50 nM T78709 CPCK60 155526570 Ki = 2860 nM T78709 C0MX4T 155526627 Ki = 66 nM T78709 C8GC1P 155526628 Ki = 0.5012 nM T78709 C1U2XO 155526651 Ki = 22 nM T78709 CXH79K 155526720 Ki = 38 nM T78709 CP76JX 155526977 Ki = 2511.89 nM T78709 C46NXV 155527302 Ki = 24.1 nM T78709 C6BHY8 155527304 Ki = 102 nM T78709 C3PS9Z 155527787 Ki = 290 nM T78709 CEQ8O4 155527891 Ki = 135 nM T78709 CL6XH7 155528009 Ki = 236 nM T78709 CIO6V1 155528183 Ki = 181.97 nM T78709 CHJ79N 155528236 Ki = 222 nM T78709 CRA6L0 155528255 Ki = 183 nM T78709 CW68KC 155528355 Ki > 10000 nM T78709 C7C1EF 155528967 Ki = 46 nM T78709 C7FR8Y 155529117 Ki = 11.48 nM T78709 C5J7AU 155529153 Ki = 5311 nM T78709 CF2DM6 155529314 Ki = 1.349 nM T78709 C9KS5C 155529450 Ki = 25 nM T78709 CEN90X 155529453 Ki = 125 nM T78709 CKZ25Y 155529679 Ki = 156 nM T78709 CD0C5A 155529797 Ki = 25 nM T78709 CGA7H6 155530006 Ki = 1074 nM T78709 C5T1OG 155530093 Ki = 239 nM T78709 C3X4IA 155530328 Ki = 21 nM T78709 C9PC3D 155530350 Ki = 989 nM T78709 C12AMJ 155530737 Ki = 321 nM T78709 CVLC03 155530779 Ki = 91 nM T78709 C98YQF 155531012 Ki = 54 nM T78709 C4W6VC 155531065 Ki = 292 nM T78709 C3ZL2V 155531279 Ki = 20.42 nM T78709 C5HWP4 155531362 Ki > 10000 nM T78709 CXOT20 155531661 Ki = 40 nM T78709 CKDE38 155531753 Ki = 1 nM T78709 C9YMR2 155531801 Ki = 194 nM T78709 CCT8V9 155531846 Ki = 8726 nM T78709 CLZY37 155531982 Ki = 24.1 nM T78709 CE3T7O 155532050 Ki = 52 nM T78709 C05KFL 155532137 Ki = 964 nM T78709 C3R4YM 155532148 Ki = 5.012 nM T78709 CS0L4A 155532204 Ki = 476 nM T78709 CX35QS 155532545 Ki > 10000 nM T78709 C3MXL6 155532834 Ki = 0.7762 nM T78709 CX6DV4 155533028 Ki = 9473 nM T78709 CTU64O 155533099 Ki = 7.244 nM T78709 C23GDV 155533534 Ki = 13 nM T78709 C3OEH2 155533648 Ki = 373 nM T78709 CZA89B 155533824 EC50 = 27.7 nM T78709 CY01GZ 155533850 Ki = 30 nM T78709 C3L0CP 155534184 Ki = 15 nM T78709 CG85SB 155534301 Ki = 94 nM T78709 CG8Y7W 155534312 Ki = 856 nM T78709 CSE59K 155534331 Ki = 336 nM T78709 C3VGT0 155534362 Ki = 42 nM T78709 CW7SV9 155534575 Ki = 24 nM T78709 CVWX57 155534647 Ki = 69 nM T78709 C8R2TB 155534729 Ki = 143.2 nM T78709 C75FSY 155534794 Ki > 10000 nM T78709 CTO4S9 155534839 Ki = 8.4 nM T78709 CU3YE7 155534933 Ki = 75.86 nM T78709 C6KF4E 155535154 Ki = 52 nM T78709 C1E7OC 155535162 Ki = 259 nM T78709 CGZ5T8 155535272 Ki = 37 nM T78709 C35NRU 155535386 Ki = 700 nM T78709 C8O4IQ 155535827 Ki = 17 nM T78709 C14JEX 155535878 Ki > 10000 nM T78709 C7YNR9 155535901 Ki = 142 nM T78709 CB79ZW 155536080 Ki = 630.96 nM T78709 C5I1JA 155536087 Ki = 12 nM T78709 CHMV76 155536112 Ki = 136 nM T78709 C72FLG 155536152 Ki = 1610 nM T78709 CQG68A 155536202 Ki = 60.26 nM T78709 CW2SC8 155536533 Ki = 40.4 nM T78709 CLZ01I 155536626 Ki = 132 nM T78709 CTB93R 155536809 Ki = 1684 nM T78709 C6LVS4 155536841 Ki = 122 nM T78709 C7FVE8 155537034 Ki = 220 nM T78709 C36FRH 155537074 Ki = 732 nM T78709 C6CFE2 155537427 Ki = 261 nM T78709 C1T8XW 155537724 Ki = 23 nM T78709 CVS04L 155537788 Ki = 369 nM T78709 CQ0WD1 155537995 Ki = 1780 nM T78709 CB8IC7 155538144 Ki = 3311 nM T78709 C5F2GI 155538236 Ki = 27 nM T78709 COYG20 155538350 Ki = 45 nM T78709 C9TIU2 155538367 Ki = 1698 nM T78709 CYC1P3 155538451 Ki = 28 nM T78709 CM08NT 155538716 Ki > 10000 nM T78709 CQ69UA 155538814 Ki = 7505 nM T78709 C0Q5NT 155538877 Ki = 489 nM T78709 CC89JF 155539461 Ki = 209 nM T78709 CAT98F 155539483 Ki = 7 nM T78709 C70SWG 155539596 Ki = 102 nM T78709 C6S8BA 155539600 Ki = 3384 nM T78709 CV9KY1 155539925 Ki = 204.1 nM T78709 C42GUK 155540147 Ki > 10000 nM T78709 C1X0IO 155540198 Ki = 350 nM T78709 C9J3BQ 155540635 Ki = 328 nM T78709 C1KA8C 155540755 Ki = 13.4 nM T78709 CR2K1T 155540795 Ki > 10000 nM T78709 CNU92V 155540807 Ki = 6.3 nM T78709 CUY87S 155540823 Ki = 15.2 nM T78709 COS2E7 155541072 Ki > 10000 nM T78709 C6B7QU 155541341 Ki = 333 nM T78709 C6SU1V 155541676 Ki > 10000 nM T78709 CP7UG2 155541866 Ki = 334 nM T78709 COZ46W 155541871 Ki = 43 nM T78709 CFH7K5 155542074 Ki = 724.44 nM T78709 CXCW81 155542321 Ki = 12530 nM T78709 C9FS3Y 155542461 Ki > 10000 nM T78709 C18OPI 155542619 Ki = 752 nM T78709 C9RV7W 155542678 Ki = 562 nM T78709 CT6HY4 155543250 Ki = 1230 nM T78709 C68MSK 155543653 Ki = 3438 nM T78709 C0QN3W 155543949 Ki = 48.7 nM T78709 CZ7O0A 155544139 Ki = 3584 nM T78709 CY57ZS 155544392 Ki = 139 nM T78709 C91VXF 155544397 Ki = 66.07 nM T78709 CR54LA 155544513 Ki = 3.162 nM T78709 CD84VK 155544810 Ki = 66 nM T78709 C3ZS0K 155544812 Ki = 294 nM T78709 C0YE6V 155544819 Ki = 78 nM T78709 C2XZD8 155545087 Ki = 79 nM T78709 CD39HU 155545397 IC50 > 1000 nM T78709 CI0YL8 155545625 Ki > 10000 nM T78709 CXI7S8 155545989 Ki = 50 nM T78709 C74GFO 155546189 Ki = 81 nM T78709 CCK3D7 155546303 Ki = 28 nM T78709 CH3W9N 155546350 Ki > 10000 nM T78709 C4C9NO 155546587 EC50 = 10100 nM T78709 C4UT5Z 155546595 Ki = 132 nM T78709 C98AIL 155546781 Ki = 128 nM T78709 C2KM3J 155547346 EC50 = 107 nM T78709 CD02EN 155547436 Ki = 47 nM T78709 CFL6E5 155547451 Ki = 42 nM T78709 COJ27N 155547693 Ki = 15070 nM T78709 CAT9X4 155548275 Ki > 10000 nM T78709 C87JGN 155549153 Ki > 10000 nM T78709 CGP8O5 155549315 Ki = 19 nM T78709 CXH9A8 155549493 Ki = 173.78 nM T78709 C3KXY1 155549528 Ki = 378 nM T78709 C52FRY 155549978 Ki = 20 nM T78709 C7YO2N 155550741 EC50 = 85000 nM T78709 C8HPN7 155551113 Ki = 64 nM T78709 C61IVC 155551353 Ki = 832 nM T78709 CHS71N 155551685 Ki = 58 nM T78709 CM26AV 155551704 Ki = 85 nM T78709 C6E9LK 155552054 Ki = 47 nM T78709 C3JEN6 155552089 Ki = 35.8 nM T78709 CX8JA1 155552185 Ki = 34 nM T78709 CQ48CS 155552188 Ki = 6.3 nM T78709 CA1WS9 155552212 Ki = 122 nM T78709 C38YJB 155552311 Ki = 142 nM T78709 C52FJU 155552469 Ki = 105 nM T78709 C0DQ3Z 155552695 Ki = 4400 nM T78709 C87PTM 155552707 Ki = 15 nM T78709 C92UAC 155552738 Ki = 62 nM T78709 CUXK56 155552760 Ki = 261 nM T78709 CDQ7C2 155552798 Ki = 536 nM T78709 C9XQ8H 155552820 Ki = 23.44 nM T78709 CPV35U 155552826 Ki > 10000 nM T78709 CBW52M 155553110 Ki = 486 nM T78709 CDV6B9 155554036 Ki = 5467 nM T78709 CFY5S4 155554150 Ki = 53 nM T78709 CKF75H 155554324 Ki = 181 nM T78709 CINW85 155554326 Ki = 91 nM T78709 C6ZSU3 155554462 Ki = 4389 nM T78709 C8JKT1 155555378 Ki = 16.4 nM T78709 C2E5TR 155555506 Ki = 775 nM T78709 CUNK28 155555525 Ki > 10000 nM T78709 CXM7C6 155555638 Ki = 246 nM T78709 C4LOH3 155555858 Ki = 15.49 nM T78709 CYP63A 155556311 Ki = 243 nM T78709 CO52HW 155556527 Ki > 10000 nM T78709 CO3G4A 155556672 Ki = 147 nM T78709 C1N5VF 155556756 Ki > 10000 nM T78709 C27JYZ 155556785 EC50 > 100000 nM T78709 CJCL47 155556806 Ki = 102 nM T78709 C5QYS0 155557134 Ki = 48 nM T78709 CXN47Z 155557425 Ki = 214 nM T78709 CD2L3K 155557443 Ki = 200 nM T78709 C8EM5K 155557592 Ki = 376 nM T78709 C0CV6O 155557695 Ki = 4.571 nM T78709 C2L0PC 155557720 Ki = 7 nM T78709 C3UCM2 155557792 Ki = 3.981 nM T78709 C9LA1I 155558180 EC50 > 500000 nM T78709 CF6H3V 155558408 Ki = 7688 nM T78709 C4I2OY 155558563 Ki = 2.1 nM T78709 C20QMI 155558704 Ki = 54.95 nM T78709 C4AG0H 155558726 Ki = 420 nM T78709 C9TB5D 155559092 Ki = 302 nM T78709 CI3G0A 155559625 Ki = 176 nM T78709 CE0HN5 155559841 Ki = 97.72 nM T78709 C3Y4RD 155560781 EC50 > 100000 nM T78709 COG70U 155560942 Ki > 10000 nM T78709 C75RMN 155561496 Ki = 1.2 nM T78709 C2HF6P 155561581 Ki = 3176 nM T78709 COL7N8 155561901 Ki = 263 nM T78709 CL45NV 155561914 Ki = 599 nM T78709 CJ57BI 155561978 Ki = 53 nM T78709 C0SDZ8 155561990 IC50 = 500 nM T78709 CW7M1D 155561995 Ki = 31 nM T78709 C8ZKT3 155562124 Ki = 1.862 nM T78709 C93KWN 155562202 Ki = 20 nM T78709 CO3C6L 155562423 Ki > 10000 nM T78709 C5AI0S 155562519 Ki = 4.9 nM T78709 C5BQ8U 155562652 Ki = 62 nM T78709 CF6B4W 155562834 Ki = 35 nM T78709 CZ6IA2 155562918 Ki = 14160 nM T78709 CYD62V 155562962 Ki = 281 nM T78709 CRCW25 155562997 Ki = 13 nM T78709 C71MOD 155563001 Ki = 1.995 nM T78709 CGC8W7 155563143 Ki = 80 nM T78709 CBH14K 155563164 Ki > 10000 nM T78709 CV9O7W 155563205 Ki > 5000 nM T78709 CG1L8E 155563286 Ki > 10000 nM T78709 C38WXS 155563374 Ki = 2467 nM T78709 C0INS4 155563826 Ki > 10000 nM T78709 CK0IW3 155563911 Ki = 37 nM T78709 C3OK2L 155565059 Ki = 160 nM T78709 CR12DI 155565189 Ki = 310 nM T78709 CQK8E3 155565209 Ki = 101 nM T78709 CE2YG1 155565215 Ki = 134 nM T78709 C3DK0P 155565218 Ki = 57.54 nM T78709 CESG75 155565298 EC50 = 11400 nM T78709 CVU9O2 155565448 Ki = 25.7 nM T78709 C19PZX 155565707 Ki = 213.8 nM T78709 CJ61GD 155565772 Ki = 257 nM T78709 C2MIU5 155565813 Ki = 202 nM T78709 C9C6WD 155565990 EC50 = 2200 nM T78709 C7P5VG 155566191 Ki = 120 nM T78709 C0D8ZO 155566396 Ki = 157 nM T78709 C5KDA9 155566405 Ki = 35.8 nM T78709 C7O6YP 155566439 Ki = 28510 nM T78709 C67LAG 155566854 Ki > 10000 nM T78709 CW1TN7 155566925 Ki = 1072 nM T78709 CRX52O 155567200 Ki = 1.622 nM T78709 C41UWT 155567307 Ki = 22 nM T78709 CBJ7M2 155567312 Ki = 50 nM T78709 CA8OE0 155567476 Ki = 2306 nM T78709 CC06FO 155567938 Ki = 38.7 nM T78709 CA68TK 155568224 Ki = 1680 nM T78709 C4EX7C 155568246 Ki = 2.3 nM T78709 C4POS3 155568373 Ki = 33.5 nM T78709 C67MIN 155568606 Ki = 0.2 nM T78709 CV5H3F 155568689 Ki = 320 nM T78709 CXP3E4 155568794 Ki = 146 nM T78709 CB5IP9 155569021 Ki = 161 nM T78709 C0CZK6 155569337 Ki > 10000 nM T78709 CP9V7M 155569396 Ki = 4365 nM T78709 C3ZNX6 155569414 Ki = 13 nM T78709 CZ8RV4 155569568 Ki = 218 nM T78709 C3N9VU 10251906 Ki > 500 nM T78709 CP9TR0 10324985 EC50 = 0.01 nM T78709 CQ1LV7 135508617 Ki = 527 nM T78709 CRKP76 136016509 Ki = 3215 nM T78709 C9J5HY 16105548 Ki = 16 nM T78709 C4ZD3A 16105549 Ki = 21 nM T78709 CFMK68 3246545 Ki = 64 nM T78709 CB2VD8 44241743 Ki = 1480 nM T78709 C13REG 44471685 Ki = 93.5 nM T78709 D00AVR 135476741 Ki > 10000 nM T78709 D00DEH 45483512 Ki = 5 nM T78709 D00FMX 46230706 Ki = 60 nM T78709 D00GSD 25107716 Ki = 188 nM T78709 D00HCC 12996705 Ki = 128 nM T78709 D00KRQ 23113096 Ki = 63 nM T78709 D00OBS 44559159 Ki > 10000 nM T78709 D00VHW 11152527 Ki = 226 nM T78709 D00YEB 25141414 Ki = 11.9 nM T78709 D01CGM 3033677 Ki = 1570 nM T78709 D01HRV 9847194 IC50 = 66 nM T78709 D01JXM 46222048 Ki > 1000 nM T78709 D01KAX 135453290 Ki = 141 nM T78709 D01KVG 9843179 Ki = 169 nM T78709 D01MBF 45483536 Ki = 156 nM T78709 D01TSX 9840090 Ki = 0.65 nM T78709 D01WWC 16573 Ki = 85 nM T78709 D01YNZ 45483529 Ki = 121 nM T78709 D02NNS 9845181 Ki = 300 nM T78709 D02RAY 16754 Ki = 171 nM T78709 D02UWB 1809 IC50 = 0.2951 nM T78709 D02YSX 197033 Ki > 100 nM T78709 D03DET 10287730 Ki = 316.23 nM T78709 D03DLZ 6089 Ki = 410 nM T78709 D03DQQ 45375938 Ki = 21 nM T78709 D03JOX 11311147 IC50 > 10000 nM T78709 D03LDH 10758200 Ki = 20.7 nM T78709 D03PYX 1219 Ki = 47 nM T78709 D03TDN 1342 Ki = 9.2 nM T78709 D03TSY 24825775 Ki = 700 nM T78709 D03XAE 10775128 Ki = 15 nM T78709 D03ZHB 44455973 Ki = 1081 nM T78709 D04AQE 1833 Ki = 3.2 nM T78709 D04DLR 128018 Ki = 842 nM T78709 D04JZJ 2838196 Ki = 120 nM T78709 D04LWD 11336800 Ki > 1000 nM T78709 D04NDO 45483400 Ki = 47 nM T78709 D04NKQ 22599992 Ki = 117 nM T78709 D04TPO 16006492 Ki = 192 nM T78709 D04TQF 11973927 Ki = 5000 nM T78709 D04TWX 9794475 IC50 > 20000 nM T78709 D04ZMS 11773145 Ki = 260 nM T78709 D04ZPF 45483409 Ki = 57 nM T78709 D05CGI 11245709 Ki = 297 nM T78709 D05EQG 5265 Ki = 17.2 nM T78709 D05GDP 599482 Ki > 10000 nM T78709 D05LJC 45483405 Ki = 606 nM T78709 D05XGR 6918647 Ki = 251.19 nM T78709 D05ZUX 44207909 Ki >= 1000 nM T78709 D06BWZ 68678 Ki = 430 nM T78709 D06DSX 12304178 Ki = 6000 nM T78709 D06FWM 44433247 Ki = 78.4 nM T78709 D06QGD 11357862 IC50 > 10000 nM T78709 D06QKW 2765 Ki = 34.67 nM T78709 D06UDU 45483520 Ki > 4570 nM T78709 D06VDN 443391 IC50 > 1000 nM T78709 D07DWS 45483446 Ki = 31 nM T78709 D07GQP 11477180 Ki = 85.4 nM T78709 D07LRJ 5312149 Ki = 340 nM T78709 D07ROK 44433248 Ki = 94.3 nM T78709 D07ZOP 11470616 IC50 > 10000 nM T78709 D08BCF 5011 Ki = 230 nM T78709 D08CKM 9863250 Ki = 1000 nM T78709 D08DOG 25130235 Ki = 42 nM T78709 D08EFH 36906 Ki = 4.6 nM T78709 D08JLB 45483406 Ki = 364 nM T78709 D08OFG 11177588 Ki > 10000 nM T78709 D08UQU 24766199 Ki = 258 nM T78709 D08VGJ 9904281 Ki = 1080 nM T78709 D08VUQ 10422832 Ki = 5.16 nM T78709 D09BNS 439280 Ki = 0.91 nM T78709 D09CKI 3037997 EC50 > 100000 nM T78709 D09HJL 10331436 IC50 > 10000 nM T78709 D09IIH 45483459 Ki = 20 nM T78709 D09MGF 11973811 Ki = 5000 nM T78709 D09OYA 2107 Ki = 12 nM T78709 D09PIN 3378093 Ki > 1000 nM T78709 D09RPR 16737207 Ki > 10000 nM T78709 D09WIL 10028436 Ki = 250 nM T78709 D0A7AK 11973810 Ki = 5000 nM T78709 D0C3EX 1797 Ki = 315 nM T78709 D0C5GF 6918515 Ki = 1470 nM T78709 D0C5XQ 1832 IC50 = 15 nM T78709 D0CA9H 25107518 Ki = 161 nM T78709 D0CG2Y 44133490 Ki = 101 nM T78709 D0CK9K 6918513 Ki = 170 nM T78709 D0DP8I 132266 Ki < 1000 nM T78709 D0E1PL 9865384 EC50 = 23.44 nM T78709 D0E3AL 56597938 Ki = 0.6 nM T78709 D0E6PQ 45483451 Ki = 128 nM T78709 D0F0IA 11301655 Ki = 1365 nM T78709 D0F6CD 5202 EC50 = 0.5 nM T78709 D0F6GB 44133853 Ki = 16 nM T78709 D0FF6S 16038374 IC50 = 10000 nM T78709 D0FU5E 10220053 Ki > 770 nM T78709 D0G2CP 10404144 Ki = 1400 nM T78709 D0G8CV 9954003 Ki = 5.012 nM T78709 D0H2TS 45483528 Ki > 1000 nM T78709 D0H3KU 172267 Ki = 344 nM T78709 D0H3WJ 44435193 Ki = 1100 nM T78709 D0H7PC 6918553 Ki > 6309.57 nM T78709 D0H9QG 5312148 Ki > 3000 nM T78709 D0I9KV 11220599 IC50 > 10000 nM T78709 D0IC4J 45375937 Ki = 11 nM T78709 D0J2UA 135433933 Ki > 10000 nM T78709 D0K3UL 9796720 Ki = 200 nM T78709 D0K6XD 44433256 Ki = 1772 nM T78709 D0K6ZT 44133851 Ki = 13 nM T78709 D0KT2M 44133674 Ki = 92 nM T78709 D0L3MJ 133538 Ki > 1000 nM T78709 D0L3XU 122187 Ki = 87 nM T78709 D0L7OM 6917970 Ki > 5000 nM T78709 D0LV7U 10667433 Ki > 1000 nM T78709 D0M2ZE 6604756 Ki = 168 nM T78709 D0M3PV 133633 Ki = 6300 nM T78709 D0M3TK 45483431 Ki = 8 nM T78709 D0N2RJ 45483432 Ki = 9 nM T78709 D0O3GF 1220 Ki = 0.17 nM T78709 D0PN8D 44351692 Ki = 2.8 nM T78709 D0Q6SH 45483408 Ki > 4570 nM T78709 D0QM3E 9870500 Ki = 3.981 nM T78709 D0R3GW 10296414 Ki = 0.3162 nM T78709 D0R3TA 45483407 Ki = 77 nM T78709 D0R5WX 11220953 Ki = 11.5 nM T78709 D0RQ8R 11973809 Ki = 5000 nM T78709 D0S0XK 9863146 IC50 = 398.11 nM T78709 D0S4JT 45483466 Ki = 189 nM T78709 D0T2RY 9948320 Ki = 280 nM T78709 D0U0VH 9904242 Ki = 0.1 nM T78709 D0V0PR 45483527 Ki > 1000 nM T78709 D0V7OO 10386282 IC50 = 5.4 nM T78709 D0W2HW 6090 Ki = 47 nM T78709 D0W8YO 46230654 Ki = 4.6 nM T78709 D0X1QW 122334 Ki = 410 nM T78709 D0X4PH 11224758 Ki = 52.7 nM T78709 D0X6MT 4106 Ki = 2.2 nM T78709 D0X8LG 11243002 IC50 > 10000 nM T78709 D0X9YS 23642275 Ki = 89.7 nM T78709 D0XX2U 16006606 Ki = 32 nM T78709 D0Y0SA 135399666 EC50 = 2890 nM T78709 D0Y1YR 442793 Ki > 100000 nM T78709 D0Y5CG 45483467 Ki = 116 nM T78709 D0Y9TL 13702393 Ki = 1701 nM T78709 D0Z1OF 23643664 Ki = 60.9 nM T78709 D0Z5GR 46230818 Ki = 4.5 nM T78709 D0ZU5W 22615724 Ki = 28 nM T12499 D00STL 644241 IC50 = 108.2 nM T12499 D03MNN 11341869 IC50 = 20 nM T12499 D03ZBT 11626560 IC50 < 1 nM T12499 D04AIT 5280445 IC50 = 10 ug.mL-1 T12499 D04LVK 57379345 IC50 = 560 nM T12499 D06XXH 11511120 IC50 = 94000 nM T12499 D09KTS 24821094 IC50 = 2.85 nM T12499 D0AZ3C 5291 IC50 = 320 nM T12499 D0E6XR 3062316 IC50 = 0.4 nM T12499 D0EG1I 9926791 IC50 = 3870 nM T12499 D0K8KX 5280343 IC50 = 40 ug.mL-1 T12499 D0OB0F 5328940 IC50 = 1.3 nM T12499 D0R0MW 5329102 IC50 = 8.9 nM T12499 D0W5HK 216239 IC50 = 60 nM T12499 D02RJY 11442891 IC50 = 155 nM T12499 D02UFQ 11620908 IC50 = 2400 nM T12499 D02XNW 5494449 Ki = 80 nM T12499 D03AND 11656518 IC50 > 6000 nM T12499 D03HUX 49792852 IC50 > 10000 nM T12499 D03LWG 53235510 IC50 = 2500 nM T12499 D07EHV 44814409 IC50 > 10000 nM T12499 D07HPJ 11476171 IC50 = 5600 nM T12499 D08AOZ 86582336 IC50 = 3800 nM T12499 D08HOM 46207586 IC50 = 3 nM T12499 D08UUL 46700756 IC50 > 10000 nM T12499 D0A5MC 11712649 IC50 = 3200 nM T12499 D0CY1B 6420138 Ki = 2800 nM T12499 D0E3TC 44259 IC50 = 1.01 nM T12499 D0G5XV 135565884 IC50 = 187 nM T12499 D0H2HZ 60194098 IC50 = 3981.07 nM T12499 D0HS5V 11234052 IC50 > 2500 nM T12499 D0LF1U 5287969 IC50 = 11000 nM T12499 D0M0XB 10302451 IC50 < 4 nM T12499 D0M9QZ 11485656 IC50 = 500000 nM T12499 D0N8RV 9868037 IC50 = 22 nM T12499 D0O0LS 25141092 IC50 > 1000 nM T12499 D0O6WV 24794418 IC50 = 120 nM T12499 D0P1CV 46191454 IC50 > 10000 nM T12499 D0Q7RE 16007391 Ki = 170 nM T12499 D0Q9UX 16718576 IC50 = 209 nM T12499 D0S4JK 24771867 IC50 = 320 nM T12499 D0S5RC 3025986 IC50 > 40000 nM T12499 D0U3EP 445154 IC50 = 112000 nM T12499 D0Z4RC 24756910 IC50 = 5910 nM T12499 D0LF0O 135441202 IC50 = 140 nM T12499 D00OWF 5280953 IC50 > 250000 nM T12499 D00PWQ 3820 IC50 = 470 nM T12499 D08DBE 10344820 Ki = 116 nM T12499 D09HEV 6539952 IC50 = 15 nM T12499 D0A9KI 9863367 IC50 > 10 nM T12499 D0F8DL 176155 IC50 = 3450 nM T12499 D0T3ME 156422 IC50 = 35000 nM T12499 D0U7OU 3220 IC50 = 5 ug.mL-1 T12499 CB1VW3 1400 IC50 = 5 nM T12499 CY58BM 1880 IC50 = 80 ug.mL-1 T12499 CZM9B7 2404 IC50 > 100000 nM T12499 CZ0T5U 2948 IC50 = 17 nM T12499 C1BE5N 3799 IC50 < 10000 nM T12499 C0W4UD 3896 IC50 = 10000 nM T12499 CBPM40 4878 Ki = 0.7943 nM T12499 CAME09 8512 IC50 > 800 ug.mL-1 T12499 C73JPZ 10639 IC50 > 800 ug.mL-1 T12499 C0RTM7 11796 IC50 = 20 ug.mL-1 T12499 C7H0NX 78630 IC50 = 2909000 nM T12499 C89ZVN 125519 IC50 = 1000 nM T12499 CWVL71 152444 IC50 = 1560000 nM T12499 CA5CO8 157820 IC50 = 18000 nM T12499 CPW0V2 165521 IC50 = 4 ug.mL-1 T12499 CV7W4J 176406 IC50 < 10000 nM T12499 C08RPS 177048 IC50 = 200000 nM T12499 CYE78A 182362 IC50 = 3 ug.mL-1 T12499 C75SNM 210813 IC50 = 5000 nM T12499 C7ER4A 229016 IC50 = 100 ug.mL-1 T12499 C2F4EP 332208 IC50 > 800 ug.mL-1 T12499 C1RBE6 368070 IC50 > 2927000 nM T12499 CHQ8V9 372421 IC50 > 2000000 nM T12499 CZH37Q 375454 IC50 = 26000 nM T12499 C0DI9H 375472 IC50 = 85000 nM T12499 C0M4OG 375473 IC50 = 1000 nM T12499 CQD2L7 380855 IC50 = 150000 nM T12499 CVJQ29 380856 IC50 = 42000 nM T12499 CCZW91 380857 IC50 = 65000 nM T12499 CA4FN2 380860 IC50 = 1000 nM T12499 CQO21P 383146 IC50 = 25000 nM T12499 C4MNG8 445840 IC50 = 2300 nM T12499 CIE63B 446044 IC50 > 200000 nM T12499 C1YNB7 447721 IC50 > 20000 nM T12499 C1ZG2U 449087 IC50 > 10000 nM T12499 C9L4RP 468132 IC50 = 5000 nM T12499 CMF14P 598873 IC50 = 1500000 nM T12499 CYC75Z 622510 IC50 > 2000000 nM T12499 C4G0QI 659323 IC50 = 260000 nM T12499 CIGS25 676030 IC50 = 80 ug.mL-1 T12499 CM2NR3 676310 IC50 = 50 ug.mL-1 T12499 C2XAH3 678080 IC50 = 999000 nM T12499 CQHO31 688662 IC50 = 40 ug.mL-1 T12499 CH5JI0 688813 IC50 > 800 ug.mL-1 T12499 C2RAL3 703616 IC50 = 622000 nM T12499 C2H5IE 735037 IC50 = 20 ug.mL-1 T12499 CA30WB 735606 IC50 > 3787000 nM T12499 C0G8LW 776222 IC50 = 307000 nM T12499 CPZV35 788949 IC50 = 205000 nM T12499 CWB7K2 814765 IC50 = 3097000 nM T12499 CYQ90E 1474874 IC50 > 100000 nM T12499 C3SGW1 1490236 IC50 = 10000 nM T12499 C7B3EF 1695774 IC50 > 800 ug.mL-1 T12499 CM8EJ4 2306385 IC50 > 2775000 nM T12499 CY32QZ 2488782 IC50 = 740 nM T12499 C9IWU0 2789324 IC50 = 50000 nM T12499 CI0P2J 2814562 IC50 = 38000 nM T12499 CHGP54 3035187 IC50 = 5000 nM T12499 CIU9K1 3049109 IC50 = 2117000 nM T12499 C2LIF3 3295701 IC50 = 619000 nM T12499 CYN03Q 3684055 IC50 > 2000000 nM T12499 CQ9YE2 3758644 IC50 = 2323000 nM T12499 CM49EB 5007981 IC50 > 2000000 nM T12499 CKWU34 5058788 IC50 > 2000000 nM T12499 CU6M8E 5280457 IC50 = 193000 nM T12499 C8ELV4 5281617 IC50 = 80 ug.mL-1 T12499 CN10FM 5281793 IC50 = 23500 nM T12499 CX4F7K 5281953 IC50 = 20 ug.mL-1 T12499 CTID76 5282335 IC50 > 40000 nM T12499 C0JX4D 5317038 IC50 > 800 ug.mL-1 T12499 CNB7Q3 5328796 IC50 = 1000000 nM T12499 C4RUV5 5329453 IC50 = 300 nM T12499 COX6Q3 5339689 IC50 = 2106000 nM T12499 CF24MP 5353259 IC50 = 60 nM T12499 CBC0E8 5374802 IC50 = 1229000 nM T12499 CJ3WR2 5381920 IC50 > 800 ug.mL-1 T12499 CVU01J 5388676 IC50 = 1500000 nM T12499 C0SO6F 5388678 IC50 = 100000 nM T12499 C9RAX0 5388679 IC50 = 500000 nM T12499 CMS0G9 5388680 IC50 = 2000000 nM T12499 CUX3A5 5388744 IC50 = 2285000 nM T12499 CA2GL7 5388745 IC50 = 516000 nM T12499 CB86MY 5391140 IC50 = 10 ug.mL-1 T12499 CR8AM5 5467796 IC50 > 2530000 nM T12499 CKX8Q5 5467800 IC50 > 2530000 nM T12499 CF0MC5 5467801 IC50 = 168000 nM T12499 CM34ED 5468835 IC50 = 74000 nM T12499 CDVG95 5481246 IC50 = 30 ug.mL-1 T12499 CDK3J0 5703619 IC50 = 3.3 nM T12499 C7H9VZ 5905112 IC50 = 2175000 nM T12499 CEZP52 6263849 IC50 > 50000 nM T12499 C03WIJ 6303920 IC50 = 615000 nM T12499 C4RVA6 6440397 IC50 = 118000 nM T12499 CA31PJ 6539953 IC50 = 40 nM T12499 C64ZJA 6539954 IC50 = 40 nM T12499 CBD1H7 6539955 IC50 = 110 nM T12499 CWHY29 6539956 IC50 = 93 nM T12499 CW76RA 6539957 IC50 = 4 nM T12499 C7K1QS 6539958 IC50 = 209 nM T12499 CJ7IL2 6539959 IC50 = 3120 nM T12499 CAE95J 6539960 IC50 = 167 nM T12499 CH86XJ 6539961 IC50 = 55 nM T12499 C41FUH 6539962 IC50 = 28 nM T12499 C7M2JP 6539963 IC50 = 92 nM T12499 CS5V1C 6539964 IC50 = 31 nM T12499 C10FYS 6539966 IC50 = 10 nM T12499 CIS1T3 6539967 IC50 = 50 nM T12499 CUPQ08 6539985 IC50 = 20000 nM T12499 CMEZ23 6540005 IC50 = 4500 nM T12499 CP0XI6 6603792 IC50 < 1 nM T12499 C3R5VW 9547983 IC50 = 3 nM T12499 CRK62A 9581370 IC50 > 3316000 nM T12499 CZDR80 9584504 IC50 > 3316000 nM T12499 C6MBQ4 9794567 IC50 = 19000 nM T12499 C2OL7K 9796455 IC50 = 1400 nM T12499 C01TAH 9802700 IC50 > 30000 nM T12499 CI80BK 9803350 IC50 = 200 nM T12499 CKT18P 9803404 IC50 > 20000 nM T12499 CSM34J 9804627 IC50 = 82 nM T12499 CR3Q2J 9818899 IC50 = 19.5 nM T12499 C2QX0O 9820995 IC50 = 1500 nM T12499 C6QBF8 9823235 IC50 = 4 nM T12499 CW8V0K 9864418 IC50 > 16000 nM T12499 CIEX48 9865315 IC50 = 3 nM T12499 C23BQG 9867983 IC50 = 650 nM T12499 C7RLN5 9867984 IC50 > 20000 nM T12499 CM5Z8X 9869943 IC50 = 0.5 nM T12499 C26LCM 9883941 IC50 = 58 nM T12499 C51QNA 9883977 IC50 = 86 nM T12499 CR2B8U 9888491 IC50 = 3300 nM T12499 CXA5C8 9893493 IC50 = 5100 nM T12499 C2Y3WG 9907612 IC50 = 300000 nM T12499 CAPU15 9908247 IC50 = 23 nM T12499 C13JNB 9917853 EC50 = 10000 nM T12499 CXD2Y6 9926586 IC50 = 3800 nM T12499 CL4TW5 9926914 IC50 = 153 nM T12499 CYW49X 9927718 IC50 = 35 nM T12499 CG6A1H 9927800 IC50 = 1100 nM T12499 C4OP1L 9932917 IC50 = 1400 nM T12499 CPQ13K 9933545 IC50 > 100000000 nM T12499 CRK63X 9933645 IC50 = 0.5 nM T12499 C6BZ2C 9934106 IC50 > 10000 nM T12499 CJO47T 9948405 IC50 > 10000 nM T12499 CJP49W 9949373 IC50 = 128 nM T12499 C54ZXH 9950678 IC50 = 2 nM T12499 CD63SU 9953450 IC50 = 290 nM T12499 CS35OC 9953741 IC50 = 27 nM T12499 CFC2E6 9954769 IC50 > 30000 nM T12499 CAH50Y 9970231 IC50 = 141000 nM T12499 CA8BC2 9976589 IC50 > 2000000 nM T12499 C37GXK 9983303 IC50 = 8000 nM T12499 C48VFS 9999126 IC50 = 2 nM T12499 CV8I5X 9999342 IC50 > 10000 nM T12499 CUY0F8 10005715 IC50 > 10000 nM T12499 CRY61O 10019770 IC50 = 102 nM T12499 C91VIF 10020232 IC50 > 2000000 nM T12499 C0IA4P 10037831 IC50 = 103000 nM T12499 CXL0R8 10038606 IC50 = 106000 nM T12499 C6AYQ3 10038709 IC50 = 7400 nM T12499 CN8T1M 10041189 IC50 > 2000000 nM T12499 C7YD1X 10048045 IC50 > 25000 nM T12499 CT4M1D 10056916 IC50 = 390 nM T12499 CG4IY8 10059651 IC50 = 17000 nM T12499 CUJR40 10062694 EC50 = 5 nM T12499 CVK3F1 10066999 IC50 = 20000 nM T12499 C7ZO6S 10073515 IC50 = 7 nM T12499 C1JUF8 10073832 IC50 = 18000 nM T12499 CF1D6Y 10075240 IC50 > 12500 nM T12499 CL9D6V 10084407 IC50 = 8500 nM T12499 C8A1TH 10085171 IC50 = 382000 nM T12499 C2C1BP 10089048 IC50 > 16000 nM T12499 C9S0TC 10104347 IC50 = 100000 nM T12499 C30CJT 10126524 IC50 = 149000 nM T12499 CL25BM 10138376 IC50 = 240 nM T12499 CREM37 10151881 IC50 = 710 nM T12499 C69DHW 10158652 IC50 < 16000 nM T12499 C5QHB6 10161543 IC50 = 170 nM T12499 CG2MT8 10176710 IC50 = 203000 nM T12499 CQU0G2 10198725 IC50 = 16000 nM T12499 CQU9K5 10200651 Ki > 5400 nM T12499 CEW30I 10217590 IC50 > 5000 nM T12499 C3UDT7 10217778 IC50 > 2030000 nM T12499 CVY59N 10244533 IC50 > 200000 nM T12499 C5TQ7X 10247543 IC50 > 10000 nM T12499 CI5N9U 10248746 IC50 = 1565000 nM T12499 C97GRN 10248747 IC50 = 26 nM T12499 C6G8NR 10264200 IC50 = 123000 nM T12499 C3HF6S 10264201 IC50 = 200000 nM T12499 CF81EM 10265006 IC50 = 502000 nM T12499 C6DC8Q 10275163 IC50 = 1600 nM T12499 C7SFI1 10296883 IC50 > 10000 nM T12499 C8RD3V 10301884 IC50 = 7 nM T12499 CDP39Q 10316258 IC50 > 2000000 nM T12499 CNS2K1 10318364 IC50 > 2030000 nM T12499 C5CBF9 10320381 IC50 = 100 nM T12499 C3JXP2 10323644 IC50 > 2030000 nM T12499 COC7P1 10333957 IC50 = 56000 nM T12499 CT7PD3 10336593 IC50 > 2000000 nM T12499 C40CWN 10343123 IC50 = 3 nM T12499 CA9L0O 10351200 IC50 = 100 nM T12499 CYCM39 10355659 IC50 = 326000 nM T12499 C37AMD 10356450 IC50 = 754000 nM T12499 C4DOQ9 10356451 IC50 = 46000 nM T12499 C50RSP 10365064 IC50 = 1.7 nM T12499 C52VFK 10366780 IC50 = 3 nM T12499 CVTI82 10377245 IC50 = 487000 nM T12499 C6NLD0 10381816 IC50 = 1876000 nM T12499 CUDE45 10397980 IC50 = 100000 nM T12499 CPS79C 10402283 IC50 = 0.62 ug.mL-1 T12499 C7WEF1 10404203 IC50 > 2000000 nM T12499 CQBD84 10410849 IC50 = 144 nM T12499 CLAX64 10413508 IC50 = 600 nM T12499 CY8H6P 10413576 IC50 > 2030000 nM T12499 CP6N2J 10423146 IC50 = 328000 nM T12499 C97TUR 10426617 IC50 > 2000000 nM T12499 C7HBP6 10429593 IC50 > 10000 nM T12499 CZ68BO 10436007 IC50 > 2030000 nM T12499 CEU25H 10445729 IC50 = 223000 nM T12499 C7ENZ5 10450419 IC50 = 2.4 nM T12499 CLP71R 10466312 IC50 = 58000 nM T12499 CW23SQ 10468973 IC50 = 1621000 nM T12499 C2WQ8M 10473563 IC50 > 10000 nM T12499 C1PB3U 10475630 IC50 > 2030000 nM T12499 C7PLI5 10478569 IC50 = 500 nM T12499 CRX6F0 10479082 IC50 = 10000 nM T12499 CJ5M1D 10482445 IC50 = 100 nM T12499 CXV6B7 10598533 IC50 = 79.7 ug.mL-1 T12499 CX64KP 10862285 IC50 = 170 nM T12499 CD62RJ 10864012 IC50 = 110 nM T12499 CFW87I 10867503 IC50 > 2000000 nM T12499 C7UP2S 10871490 IC50 = 150 nM T12499 CIQ49T 10885591 IC50 = 120 nM T12499 CEJ1S7 10893387 IC50 = 380 nM T12499 CYU8L6 10893773 IC50 > 40000 nM T12499 CBTD58 10894116 IC50 > 40000 nM T12499 C9AYL4 10909252 IC50 > 50000 nM T12499 CSU61K 10916861 IC50 = 730 nM T12499 CUZ74A 10928594 IC50 > 40000 nM T12499 CL9RB3 10939823 IC50 = 740 nM T12499 C8T7AZ 10948261 IC50 = 11000 nM T12499 CLU1O8 10950004 IC50 = 2 nM T12499 CZOF70 10951171 IC50 = 4 nM T12499 C7YX3I 10961937 IC50 = 30 nM T12499 C3C5EL 10962019 IC50 = 2000 nM T12499 CF9IZ1 10970293 IC50 > 40000 nM T12499 CT2N0F 10975200 IC50 = 33800 nM T12499 C0B6ZI 10979411 IC50 = 26000 nM T12499 CM8T6S 10981996 IC50 > 40000 nM T12499 CF7YV3 10982890 IC50 = 5100 nM T12499 CRZ3N4 10983330 IC50 = 2 nM T12499 C46KPJ 11003870 IC50 = 45 nM T12499 CMTX54 11014882 IC50 = 780 nM T12499 CIH8S7 11047384 IC50 = 460 nM T12499 CJ3G8F 11047824 IC50 = 18 nM T12499 CJV52R 11048780 IC50 = 460 nM T12499 C5MBH4 11051416 IC50 > 50000 nM T12499 CP0DG3 11058515 IC50 = 770 nM T12499 CP15QT 11060735 IC50 = 600 nM T12499 C91ZML 11070550 IC50 = 360 nM T12499 CK09XA 11073138 IC50 = 5020 nM T12499 C18KEF 11078754 IC50 > 40000 nM T12499 CPME05 11079939 IC50 = 9600 nM T12499 CO8H4W 11089354 IC50 = 460 nM T12499 C8GE1S 11090362 IC50 = 9600 nM T12499 CRY3O4 11091267 IC50 = 570 nM T12499 C96EUC 11111399 IC50 = 770 nM T12499 CIK0Z6 11113249 IC50 = 86 nM T12499 CE9W7F 11114178 IC50 = 10 nM T12499 C1R2VS 11123387 IC50 = 26 nM T12499 CN1CJ5 11124103 IC50 = 440 nM T12499 C97ISW 11134621 IC50 = 2 nM T12499 C03JWT 11135291 IC50 = 180 nM T12499 CFBH56 11144210 IC50 = 5900 nM T12499 C7I4RG 11147222 IC50 = 3800 nM T12499 CN2JQ0 11169051 IC50 = 23 nM T12499 CS9CK8 11186472 IC50 > 50000 nM T12499 CH3P1J 11186612 IC50 = 4800 nM T12499 CD9E2W 11188787 IC50 = 8 nM T12499 C0Y8TX 11192751 IC50 = 8 nM T12499 CEUR60 11192985 IC50 = 6 nM T12499 CBF04J 11197310 IC50 > 2000000 nM T12499 CO6K3J 11200510 IC50 < 0.2 nM T12499 CB06ZF 11204217 IC50 = 19 nM T12499 CT3K9Z 11213588 IC50 = 1 nM T12499 CEJ6F2 11214762 IC50 = 20 nM T12499 C4HUM2 11232168 IC50 = 10000 nM T12499 C2W5RC 11235063 IC50 > 50000 nM T12499 CVOW82 11238420 IC50 = 210 nM T12499 C02GWO 11245369 IC50 > 30000 nM T12499 CWD28N 11256035 IC50 > 50000 nM T12499 C8JK6G 11257376 IC50 = 98000 nM T12499 CLCW19 11260009 IC50 = 0.7 nM T12499 CC2L8U 11268003 IC50 > 50000 nM T12499 CNBX16 11270660 IC50 = 8 nM T12499 CEP0G1 11273105 IC50 = 10 nM T12499 C2HA7W 11283174 IC50 = 0.5 nM T12499 CBOP58 11293798 Ki > 10000 nM T12499 C9S8PK 11295293 IC50 = 96 nM T12499 CXS5E4 11316381 IC50 = 87 nM T12499 CGP80V 11328586 IC50 = 188 nM T12499 CDI42Q 11328827 IC50 < 0.5 nM T12499 CU5P8C 11331007 IC50 = 12 nM T12499 CC38HS 11336689 IC50 = 8.7 nM T12499 CW0JF9 11337764 IC50 = 121000 nM T12499 CEC31B 11351900 IC50 = 63 nM T12499 C0J2TB 11359024 IC50 = 10000 nM T12499 CFQ7J6 11361039 IC50 = 28000 nM T12499 C26BZX 11362471 Ki > 10000 nM T12499 CB45PJ 11362483 IC50 = 1200 nM T12499 C9B4XP 11363872 IC50 = 4 nM T12499 CGN8P2 11365768 IC50 = 6 nM T12499 C43NPS 11373886 IC50 > 10000 nM T12499 CP4ZO0 11375301 IC50 = 20 nM T12499 CT6Y9W 11376799 IC50 = 23 nM T12499 CEAR81 11381572 IC50 > 50000 nM T12499 CM30TC 11387552 IC50 = 240 nM T12499 CG9Y8F 11395429 IC50 = 5800 nM T12499 CWXB93 11397177 Ki > 10000 nM T12499 CV2IN9 11404920 IC50 = 10000 nM T12499 CMA4U9 11407465 IC50 = 0.2 nM T12499 CYW65I 11417763 IC50 = 380 nM T12499 C73PUW 11420344 IC50 = 18 nM T12499 C5O1RM 11421633 IC50 = 5 nM T12499 C71PYD 11427975 IC50 = 22000 nM T12499 C7AI2V 11432911 IC50 = 7800 nM T12499 C3AS8V 11439407 IC50 > 50000 nM T12499 CYD2A6 11440253 IC50 = 370 nM T12499 CFJ6B2 11441375 IC50 = 330 nM T12499 CO4F0R 11443738 IC50 = 350 nM T12499 CKM8E6 11444953 IC50 = 10 nM T12499 CJC95A 11454205 IC50 > 10000 nM T12499 CU50OG 11455909 IC50 = 12 nM T12499 CFN2C0 11466196 IC50 = 0.7 nM T12499 C4Q7XD 11474276 IC50 = 300 nM T12499 C6M9NC 11477626 IC50 = 4700 nM T12499 CDOF16 11484790 IC50 = 1900 nM T12499 C2Z7WP 11486459 IC50 = 1200 nM T12499 CLM98C 11487256 IC50 = 0.5 nM T12499 CPC9S5 11489476 IC50 = 190 nM T12499 C0H6QS 11495680 IC50 > 10000 nM T12499 C8RQD7 11501591 IC50 = 122 nM T12499 CIW9L5 11502867 IC50 > 10000 nM T12499 CU2OF8 11510392 IC50 = 0.6 nM T12499 C2T8YD 11511361 IC50 = 860 nM T12499 CK2Q0X 11516978 IC50 > 10000 nM T12499 C8AY3B 11518031 IC50 < 25 nM T12499 C87ARG 11519208 IC50 = 170 nM T12499 CHW13Q 11519350 IC50 = 8 nM T12499 CO70EZ 11526166 IC50 = 1480 nM T12499 CPE53F 11526238 IC50 > 10000 nM T12499 C7HMO6 11526786 IC50 > 30000 nM T12499 C5BM4T 11531799 IC50 > 10000 nM T12499 C53OSD 11532048 IC50 > 10000 nM T12499 CC4QM5 11532676 IC50 > 10000 nM T12499 C05FSE 11538753 IC50 = 35 nM T12499 CTG83F 11539329 Ki > 2700 nM T12499 CN1K3R 11545702 IC50 = 1 nM T12499 C01FVM 11546457 IC50 > 10000 nM T12499 C32PUD 11553058 IC50 = 210 nM T12499 CW43OA 11554885 IC50 = 14 nM T12499 CACS26 11561968 Ki > 2000 nM T12499 CNBM81 11562171 IC50 > 10000 nM T12499 CJ59WD 11562553 IC50 = 14 nM T12499 C9XI8Z 11574885 IC50 = 30 nM T12499 CO9KP5 11583459 IC50 > 10000 nM T12499 CA2KX0 11590078 IC50 = 11700 nM T12499 CMIL86 11590363 Ki > 2700 nM T12499 C3CS5K 11593704 IC50 > 3787000 nM T12499 C0NV9Y 11596881 IC50 > 10000 nM T12499 C45BMY 11603130 IC50 = 2100 nM T12499 C69FYK 11604142 Ki = 400 nM T12499 COW68T 11605551 IC50 > 100000 nM T12499 CU6T2L 11613133 IC50 = 30 nM T12499 C1BLZ5 11620055 IC50 > 10000 nM T12499 CUO43M 11620207 IC50 > 25000 nM T12499 CUQ4I5 11620266 IC50 = 27 nM T12499 C5B3XJ 11620410 IC50 = 1140 nM T12499 CG1JN5 11620467 IC50 = 54 nM T12499 C70LDZ 11625929 IC50 < 1 nM T12499 C9ZD2E 11626406 IC50 = 36 nM T12499 CX72ET 11626681 IC50 = 83 nM T12499 CPB48V 11626947 IC50 = 42 nM T12499 CWM80X 11627419 IC50 = 210 nM T12499 CK34LS 11632737 IC50 > 50000 nM T12499 CYL45U 11634544 IC50 = 200 nM T12499 C7CV8O 11634876 IC50 = 22 nM T12499 C1TZY3 11635079 IC50 = 22 nM T12499 C9T6SC 11640926 Ki > 2700 nM T12499 CVH29N 11642023 IC50 = 1920 nM T12499 CA80WI 11648745 IC50 = 11 nM T12499 C82TKN 11656437 IC50 = 11 nM T12499 C3L2HT 11656560 IC50 = 380 nM T12499 CX7C1T 11656606 IC50 = 29 nM T12499 C1AUX0 11661290 IC50 = 36 nM T12499 C24GRQ 11661959 IC50 > 10000 nM T12499 C60ASI 11663230 Ki = 138 nM T12499 C8RMT2 11663885 IC50 = 19 nM T12499 CCGO58 11669282 IC50 = 154 nM T12499 C1LV6H 11677453 IC50 = 11 nM T12499 CA4Q5F 11678465 IC50 = 22 nM T12499 CS72ED 11682843 IC50 > 10000 nM T12499 C5O6YX 11683692 IC50 = 0.4 nM T12499 CP3U0W 11684933 IC50 = 9 nM T12499 CYO6X9 11684994 Ki = 138 nM T12499 CCEY64 11689855 IC50 = 65 nM T12499 CU0E8O 11690457 Ki > 2000 nM T12499 CLC53E 11691173 IC50 > 10000 nM T12499 CI3EO4 11692100 IC50 = 1600 nM T12499 CB0AP2 11705863 Ki > 2000 nM T12499 C6EUQ9 11711497 IC50 = 10 nM T12499 C9ROB0 11713267 IC50 = 21 nM T12499 C1FTX3 11719305 IC50 > 10000 nM T12499 CZY05V 11719421 IC50 = 13 nM T12499 CQN04F 11723994 IC50 > 2000000 nM T12499 C0NVT9 11724908 IC50 > 2000000 nM T12499 C6N2AQ 11726550 IC50 = 2 nM T12499 CX21FQ 11727911 IC50 = 27 nM T12499 CGA26L 11729126 IC50 = 2500 nM T12499 C84LGZ 11730798 IC50 = 50 nM T12499 CA9HO6 11730954 IC50 = 120 nM T12499 CT7U6H 11731262 IC50 = 25 nM T12499 CPY1Z2 11740563 IC50 = 290 nM T12499 CS5QL4 11749561 IC50 = 700 nM T12499 CN8S1E 11752715 IC50 = 28 nM T12499 CE0KI4 11753519 IC50 = 110 nM T12499 CP7AH3 11755812 IC50 = 50000 nM T12499 CUKE53 11760559 IC50 = 1100 nM T12499 CMJ2Q9 11761204 IC50 > 2500 nM T12499 C28UON 11775143 IC50 = 1.3 nM T12499 C3J7MT 11777791 IC50 = 117000 nM T12499 C96TSA 11784426 IC50 = 2500 nM T12499 CL87KR 11785748 IC50 = 27 nM T12499 CCI6R5 11842847 IC50 = 1 nM T12499 CMO6N4 11842849 IC50 = 13 nM T12499 C9HT7B 11842850 IC50 = 49 nM T12499 CP6KY2 11843009 IC50 = 1 nM T12499 C8FHK9 11843010 IC50 = 1 nM T12499 C7D6MQ 11843012 IC50 = 1 nM T12499 C4T2WC 11843013 IC50 = 1 nM T12499 CS36BH 11843159 IC50 = 0.6 nM T12499 C7DU6T 11843160 IC50 = 2 nM T12499 CH6W3V 11844349 IC50 = 14 nM T12499 CI15NA 11844350 IC50 = 12 nM T12499 CUL2C8 11844485 IC50 = 10 nM T12499 C96ORQ 11844486 IC50 = 1 nM T12499 C4SK3L 11844487 IC50 = 1 nM T12499 C6KF8Z 11844488 IC50 = 1 nM T12499 C9ECK3 11844489 IC50 = 1 nM T12499 C83YRX 11844616 IC50 = 1 nM T12499 CV24WL 11844764 IC50 = 1 nM T12499 C9JT4S 11847343 IC50 > 10000 nM T12499 CAZS08 11848309 IC50 = 3614 nM T12499 C43IVN 11848567 IC50 = 1335 nM T12499 C9LAY8 11848825 IC50 > 10000 nM T12499 CHR92S 11858109 IC50 < 4 nM T12499 CHN2X6 11974313 IC50 = 3200 nM T12499 CTN38E 11974315 IC50 = 124 nM T12499 COFI19 11974316 IC50 = 47 nM T12499 CU4IJ6 12035491 IC50 = 700 nM T12499 CA4Z6H 12373545 IC50 > 2916000 nM T12499 C8YVD5 12381316 IC50 > 2000000 nM T12499 C5CPV2 12516472 IC50 > 10 ug.mL-1 T12499 CS0Y1J 12634029 IC50 = 18500 nM T12499 C1PI2A 12911686 IC50 > 50000 nM T12499 CU4C3V 12968172 IC50 = 11 nM T12499 CI8VE5 12968173 IC50 = 2290 nM T12499 CR75GZ 12968174 IC50 = 260 nM T12499 CEVY69 12968175 IC50 = 4 nM T12499 CL1PR6 12968176 IC50 = 17 nM T12499 CY5EA7 12968177 IC50 = 470 nM T12499 CZ98FV 12968178 IC50 = 310 nM T12499 C4SUK6 12968179 IC50 = 144 nM T12499 CGIZ84 12968180 IC50 = 20 nM T12499 C5MX8N 12968181 IC50 = 30 nM T12499 C0P5HT 13182760 IC50 > 800 ug.mL-1 T12499 CS6FK7 14304977 IC50 > 2000000 nM T12499 CQ29NJ 14304982 IC50 > 2000000 nM T12499 CA8E6W 14791361 IC50 = 1160000 nM T12499 CRED76 14791362 IC50 > 2000000 nM T12499 C8ZS9R 14791363 IC50 > 2000000 nM T12499 CH5RB9 14791364 IC50 > 2000000 nM T12499 C5UD8T 14791365 IC50 > 2000000 nM T12499 C25VAZ 14791366 IC50 > 2000000 nM T12499 CES4B9 14791367 IC50 > 2000000 nM T12499 C8R3IO 14791368 IC50 > 2000000 nM T12499 CLOA14 14791369 IC50 > 2000000 nM T12499 C9HLZ3 14791370 IC50 > 2000000 nM T12499 C5N6QA 14791371 IC50 > 2000000 nM T12499 CNB0F4 14791372 IC50 > 2000000 nM T12499 CM87DK 14791373 IC50 > 2000000 nM T12499 CR0J2L 14791374 IC50 > 2000000 nM T12499 CP2H9Y 14791375 IC50 > 2000000 nM T12499 CLXA81 14791376 IC50 > 2000000 nM T12499 CN3F5B 14791377 IC50 > 2000000 nM T12499 CRK9U6 14791378 IC50 > 2000000 nM T12499 CQ5F7V 14791379 IC50 > 2000000 nM T12499 C3RNU7 14791380 IC50 = 1595000 nM T12499 CI98LS 14791381 IC50 = 1032000 nM T12499 C9S7KU 14791382 IC50 = 439000 nM T12499 CWAV76 14791383 IC50 > 2000000 nM T12499 CGX9C2 14791384 IC50 > 2000000 nM T12499 C2YW0J 14791386 IC50 > 2000000 nM T12499 CM3Q7F 14791387 IC50 = 810000 nM T12499 CG10QR 14791388 IC50 > 2000000 nM T12499 C49FJH 14791389 IC50 > 2000000 nM T12499 CX8R7N 14791390 IC50 > 2000000 nM T12499 C0PRG2 14791391 IC50 > 2000000 nM T12499 CZ6WJ9 14791392 IC50 = 100000 nM T12499 CQ9Z0L 15550318 IC50 = 1200 nM T12499 CR7QG2 15550584 IC50 = 144 nM T12499 CF9S5H 15664638 IC50 = 234000 nM T12499 CARI31 15693660 IC50 = 40 ug.mL-1 T12499 CP9CD6 15693661 IC50 = 400 ug.mL-1 T12499 CDSL43 15693662 IC50 = 40 ug.mL-1 T12499 CWO05F 15693663 IC50 > 800 ug.mL-1 T12499 CER56U 15693664 IC50 = 40 ug.mL-1 T12499 C2Z1FO 15693665 IC50 = 40 ug.mL-1 T12499 CLG0Z7 15693666 IC50 = 200 ug.mL-1 T12499 CD7K9N 15693667 IC50 = 70 ug.mL-1 T12499 C0YWD7 15693668 IC50 > 800 ug.mL-1 T12499 C9M0SA 15693669 IC50 > 800 ug.mL-1 T12499 CUI6E5 15858664 IC50 = 200 nM T12499 CG07CP 15931492 IC50 = 1315000 nM T12499 CU9L0Z 15931493 IC50 > 3275000 nM T12499 C0M7TW 15948947 IC50 = 238 nM T12499 C1VNB4 15948949 IC50 = 7 nM T12499 CH8ZG5 15949048 IC50 = 11 nM T12499 CKNZ36 15949147 IC50 = 2090 nM T12499 CX9GH4 15949237 IC50 = 438 nM T12499 CK2Z6Y 15949521 IC50 = 32 nM T12499 CBZF29 15949522 IC50 = 132 nM T12499 C34MCY 15949523 IC50 = 11 nM T12499 CS3P9G 15949524 IC50 = 4 nM T12499 C1KPH2 15949525 IC50 = 1162 nM T12499 C5JG9R 15949617 IC50 = 4 nM T12499 C8FT6U 15949618 IC50 = 316 nM T12499 C30PVQ 15949619 IC50 = 120 nM T12499 C3PNO2 15949620 IC50 = 18 nM T12499 C4I5RS 15949621 IC50 = 2030 nM T12499 C8JLW2 15949711 IC50 > 2500 nM T12499 CVJ9A0 15949712 IC50 = 7 nM T12499 CD9IP6 15949713 IC50 > 2500 nM T12499 C2TAW9 15949714 IC50 > 2500 nM T12499 C5RI8G 15949799 IC50 = 789 nM T12499 CEI2K8 15949887 IC50 = 31 nM T12499 CAIN63 15949888 IC50 > 2500 nM T12499 C2VDI1 15949889 IC50 = 27 nM T12499 COC02T 15949890 IC50 = 881 nM T12499 CFQ6X3 15949974 IC50 = 29 nM T12499 CMKZ23 15949975 IC50 = 111 nM T12499 CWM5L4 15949976 IC50 = 6 nM T12499 CL1HO8 15950062 IC50 = 5 nM T12499 CA8S3R 15950063 IC50 = 119 nM T12499 CZ5F0K 15950065 IC50 = 583 nM T12499 CO7NG2 15950141 IC50 = 12 nM T12499 COIG45 15950224 IC50 = 7 nM T12499 C9V0TO 15950311 IC50 = 20 nM T12499 C9RQN8 15950748 IC50 = 14 nM T12499 CSK90Y 15991573 IC50 = 0.2 nM T12499 CPNW35 15991575 IC50 = 0.5 nM T12499 CFPW41 16007116 Ki > 2700 nM T12499 C09OWB 16015442 IC50 = 531 nM T12499 C0VF7Y 16037922 IC50 = 87 nM T12499 CN36QI 16043219 IC50 = 2 nM T12499 CFKE48 16064750 IC50 = 2000 nM T12499 CIHG50 16066841 IC50 = 3 nM T12499 CBU2X4 16066842 IC50 = 867 nM T12499 C3ZV2X 16086076 IC50 = 6 nM T12499 C0SO7D 16086077 IC50 = 0.6 nM T12499 C0WU9I 16086078 IC50 = 0.07 nM T12499 CVE6C8 16086088 IC50 = 0.27 nM T12499 CH1R8K 16086091 IC50 = 0.3 nM T12499 CT4RS8 16086092 IC50 = 8 nM T12499 CZ2QU1 16086093 IC50 = 297 nM T12499 C13OVU 16086099 IC50 = 0.01 nM T12499 C2YC0S 16086100 IC50 = 0.3 nM T12499 C28UZX 16086101 IC50 = 1 nM T12499 CKM8E4 16086102 IC50 = 0.5 nM T12499 CF0N4J 16086103 IC50 = 3 nM T12499 CKR57M 16086104 IC50 = 0.5 nM T12499 CI5HJ8 16086105 IC50 = 48 nM T12499 C68SBO 16086106 IC50 = 2 nM T12499 CAYV39 16086107 IC50 = 0.4 nM T12499 C06NOI 16086108 IC50 = 2 nM T12499 C6F2YX 16086109 IC50 = 150 nM T12499 CE71TI 16086110 IC50 = 0.5 nM T12499 CQ3UF2 16086111 IC50 = 0.9 nM T12499 CFXT05 16086112 IC50 = 200 nM T12499 C16NRY 16086114 IC50 = 0.2 nM T12499 C87TPW 16086115 IC50 = 3 nM T12499 CW35LJ 16086116 IC50 = 0.4 nM T12499 CA3BD7 16086117 IC50 = 14 nM T12499 C3EKF4 16086118 IC50 = 6 nM T12499 C0QCG4 16086142 IC50 = 1 nM T12499 C73MLJ 16108977 IC50 < 1 nM T12499 CQG45C 16109001 IC50 = 1100 nM T12499 C8P4ZK 16109016 IC50 = 19 nM T12499 CY1E3Q 16109017 IC50 = 42 nM T12499 CV7S6Z 16109018 IC50 = 370 nM T12499 CB98HV 16109019 IC50 = 780 nM T12499 C49VTS 16109020 IC50 = 620 nM T12499 C6FZ7A 16109023 IC50 = 1 nM T12499 CWS8D0 16109024 IC50 = 4 nM T12499 C1WS6E 16109034 IC50 = 410 nM T12499 C8IES6 16109035 IC50 = 150 nM T12499 C1U8XW 16109036 IC50 = 130 nM T12499 CNG5L6 16109037 IC50 = 1100 nM T12499 C34KRB 16109040 IC50 = 1 nM T12499 CZ5Y3V 16116847 IC50 = 5 nM T12499 CLO43V 16116849 IC50 = 48 nM T12499 C0HO6T 16118191 IC50 = 0.6 nM T12499 CT92BZ 16118192 IC50 = 1.4 nM T12499 CIZ6B4 16118193 IC50 = 0.3 nM T12499 C2CN5O 16118323 IC50 = 1.5 nM T12499 C4GTU3 16118324 IC50 = 1.3 nM T12499 CXC78K 16118603 IC50 = 63 nM T12499 CI4E6Y 16118605 IC50 = 72 nM T12499 C8LIW4 16118609 IC50 = 24 nM T12499 CGC34R 16118737 IC50 = 0.6 nM T12499 CAN2K6 16118739 IC50 = 1310 nM T12499 C5VPH9 16129448 IC50 = 2330 nM T12499 CZ08YH 16214904 IC50 = 81 nM T12499 CP3HS4 16220354 IC50 > 50000 nM T12499 CVZK29 16223008 IC50 > 50000 nM T12499 CZO8P2 16440205 IC50 = 50000 nM T12499 C6TQ2O 16664354 Ki = 11.7 nM T12499 C0H8UN 16730109 IC50 > 50000 nM T12499 C6S3YO 16731782 IC50 = 132 nM T12499 CK9CV4 16733534 IC50 = 405 nM T12499 CDZ31W 16747696 IC50 = 30963 nM T12499 C86UEN 16897096 IC50 = 160 nM T12499 CL9BQ6 17748275 IC50 = 146 nM T12499 C28TDB 17756743 IC50 = 81 nM T12499 CWH37T 17758574 IC50 = 4500 nM T12499 CUTS51 17960401 IC50 = 9 nM T12499 C1H7BJ 18007099 IC50 = 3700 nM T12499 C1V7AK 18007100 IC50 > 12500 nM T12499 C1V8BU 18007104 IC50 > 12500 nM T12499 C0Z6RE 18332602 IC50 = 800 nM T12499 C0NKJ2 18332605 IC50 = 1260 nM T12499 CRN5K7 18332650 IC50 = 1 nM T12499 CJ3TD7 18332663 IC50 = 46 nM T12499 CFL69G 18332667 IC50 = 242 nM T12499 CX6BH1 18332672 IC50 = 11 nM T12499 C9RHI4 18342784 IC50 = 1 nM T12499 CJK36Q 18354367 IC50 = 11.8 nM T12499 CP73AB 18354386 IC50 = 26.5 nM T12499 CU83MW 18354409 IC50 > 1000 nM T12499 C5RY6O 18375493 IC50 = 827 nM T12499 CA7T2W 18450829 IC50 = 380 nM T12499 CB2LF3 18450830 IC50 > 50000 nM T12499 CW0U4Z 18450843 IC50 = 140 nM T12499 C6E4YZ 18450934 IC50 = 9650 nM T12499 C0VWB3 18451020 IC50 = 290 nM T12499 C3J5HU 18451023 IC50 = 2950 nM T12499 CJA0D6 18451024 IC50 = 190 nM T12499 C0X9RC 18451029 IC50 = 230 nM T12499 CNBP94 18451030 IC50 = 6700 nM T12499 C6FQB7 18451036 IC50 = 290 nM T12499 CEI23S 18451044 IC50 = 770 nM T12499 CUZ1E0 18451049 IC50 = 1370 nM T12499 CGT10H 18451102 IC50 = 6850 nM T12499 CM9BN5 18451119 IC50 = 1520 nM T12499 CM1X8S 18451204 IC50 = 4810 nM T12499 CB84DI 18451225 IC50 = 20800 nM T12499 C45MTJ 18451346 IC50 = 5200 nM T12499 CYJ3M1 18451394 IC50 = 720 nM T12499 CHDY96 18770788 IC50 = 50000 nM T12499 C1GAJ2 18770840 IC50 = 500 nM T12499 CHI4W7 18770845 IC50 = 5000 nM T12499 C1C0EJ 18792861 IC50 = 360 nM T12499 C6HK0S 18792868 IC50 = 400 nM T12499 C4SPG1 19007057 Ki = 2800 nM T12499 C5WAV7 19597382 IC50 = 20 nM T12499 CU5CK6 19597400 IC50 = 140 nM T12499 CZQ92B 19597433 IC50 < 1 nM T12499 C02JLX 19597448 IC50 < 3 nM T12499 CYIX85 19597450 IC50 = 8 nM T12499 CFH4I2 19597457 IC50 < 3 nM T12499 CIBE65 19597460 IC50 = 130 nM T12499 C0JQ7H 19597465 IC50 < 1 nM T12499 CP01WN 19597468 IC50 < 1 nM T12499 CA09JB 19597476 IC50 = 5 nM T12499 CC78WA 19597518 IC50 = 390 nM T12499 CV0U1N 19597532 IC50 < 3 nM T12499 C1B3DX 19597536 IC50 < 1 nM T12499 C0E2OG 20579089 IC50 = 2200 nM T12499 CIC6E2 20703609 IC50 = 0.4 nM T12499 C5BS4H 20703624 IC50 = 2.6 nM T12499 CKE9O1 20703628 IC50 = 0.25 nM T12499 CX90RK 20703629 IC50 = 75.2 nM T12499 CRCY81 20703632 IC50 = 22.5 nM T12499 C4AZQ7 20703633 IC50 > 1000 nM T12499 C58WTF 20703634 IC50 = 501 nM T12499 CC1MJ6 20711999 IC50 = 40 nM T12499 CV7C2K 20817018 IC50 = 64 nM T12499 CQ5X7V 20817081 IC50 = 20 nM T12499 CEU1O0 20817327 IC50 = 341 nM T12499 CK1TF6 20817330 IC50 = 102 nM T12499 C6AN8E 20817403 IC50 = 23 nM T12499 C56HRP 20817416 IC50 = 106 nM T12499 CXCF38 20817425 IC50 = 30 nM T12499 CC1E7R 21078798 Ki > 5400 nM T12499 CH4B5K 21081523 IC50 > 5000 nM T12499 C25UKC 21081761 IC50 = 290 nM T12499 CU29EB 21137651 IC50 = 700 nM T12499 CBTS02 21137686 IC50 > 30000 nM T12499 CI82BH 21137692 IC50 = 12500 nM T12499 CA73LU 21137693 IC50 = 4400 nM T12499 CGB54O 21774685 IC50 = 92 ug.mL-1 T12499 C9RSY1 21911223 IC50 = 4.9 nM T12499 CAO1M7 21911235 IC50 = 180 nM T12499 C0D6BH 21911241 IC50 = 4470 nM T12499 CNTX42 21911266 IC50 = 1.2 nM T12499 CF9D4B 21911267 IC50 = 3 nM T12499 CQ2U0F 21911271 IC50 = 360 nM T12499 CC3UI5 21911283 IC50 = 1340 nM T12499 CEV1N5 21911286 IC50 = 18 nM T12499 CZ2K3O 21911293 IC50 = 5 nM T12499 CB5DO1 21911296 IC50 = 12080 nM T12499 CK06DT 21911324 IC50 = 3100 nM T12499 C6RM2E 21911333 IC50 = 6.3 nM T12499 C82VPK 21911338 IC50 = 4 nM T12499 C4FWH1 21911345 IC50 = 0.6 nM T12499 CQAW69 21911406 IC50 = 240 nM T12499 CCU5P6 21911412 IC50 = 130 nM T12499 CO36ZH 21911439 IC50 = 6.7 nM T12499 C0QTP8 21911457 IC50 = 50 nM T12499 C7ICY1 21911468 IC50 = 890 nM T12499 C1PTM5 21911491 IC50 = 620 nM T12499 CJV64F 21911517 IC50 = 800 nM T12499 CW81PU 21911520 IC50 = 9.4 nM T12499 CFW5Q4 21911536 IC50 = 17 nM T12499 CPN2M4 21911557 IC50 = 140 nM T12499 CXZ3J0 21911563 IC50 = 480 nM T12499 CK8AY5 21911573 IC50 = 2230 nM T12499 C01PAE 21911582 IC50 = 130 nM T12499 C4X9VW 21911584 IC50 = 390 nM T12499 CD91KJ 21911586 IC50 = 1.2 nM T12499 CL8V5Y 21911599 IC50 = 4 nM T12499 CLP84C 21911609 IC50 = 1400 nM T12499 CQWN07 21911611 IC50 = 710 nM T12499 CU59WY 21911623 IC50 = 0.5 nM T12499 C8EA6U 21911645 IC50 = 0.3 nM T12499 CX8Z1W 21985424 IC50 = 1200 nM T12499 CDS2B9 21985432 IC50 = 30 nM T12499 CP78LH 21985486 IC50 = 1300 nM T12499 C5WHN8 21994549 IC50 > 12500 nM T12499 CCPU92 21994552 IC50 = 2.4 nM T12499 CWZ8Y4 21994558 IC50 = 180 nM T12499 CKM54W 21994560 IC50 > 12500 nM T12499 C7JX0Z 21994562 IC50 = 4390 nM T12499 CEVT05 21994569 IC50 = 3 nM T12499 C6AQD0 21994570 IC50 = 820 nM T12499 CIO8H7 21994571 IC50 = 36 nM T12499 CI9D2L 21994591 IC50 = 2680 nM T12499 C6XQ1W 21994598 IC50 = 6 nM T12499 C1RUF7 21994601 IC50 = 1690 nM T12499 CRCD41 21994605 IC50 = 15 nM T12499 CJX07Q 21994606 IC50 = 890 nM T12499 C8ZN2J 21994630 IC50 > 12500 nM T12499 C21IJA 21994643 IC50 = 9.4 nM T12499 C86ONB 21994661 IC50 = 13 nM T12499 CA8B9K 21994707 IC50 = 16 nM T12499 CF35EU 21994709 IC50 = 9 nM T12499 C98IEP 21994713 IC50 = 3 nM T12499 CDIZ08 21994718 IC50 = 390 nM T12499 CBF70N 21994727 IC50 = 2 nM T12499 CDK0B1 21994742 IC50 = 3170 nM T12499 C43XZF 21994749 IC50 = 240 nM T12499 C71VCF 21994770 IC50 = 3 nM T12499 C1RV3C 21994777 IC50 = 10 nM T12499 CPFU26 21994778 IC50 = 14 nM T12499 CZ4CB9 21994781 IC50 = 100 nM T12499 C5FR4C 21994782 IC50 = 5520 nM T12499 CJV9A0 21994783 IC50 = 30 nM T12499 CQG8B4 21994786 IC50 = 60 nM T12499 CA5L3Q 21994789 IC50 = 1 nM T12499 CV78HM 21994811 IC50 > 12500 nM T12499 CLK0T6 21994850 IC50 = 11 nM T12499 C2RTU9 21994872 IC50 > 12500 nM T12499 CKA1C7 21994883 IC50 = 4 nM T12499 CZO46G 21994907 IC50 = 30 nM T12499 C2U5YF 21994914 IC50 = 4 nM T12499 C9XDA4 21994918 IC50 > 12500 nM T12499 CSEX73 21994919 IC50 = 360 nM T12499 CEPU70 21994926 IC50 = 9 nM T12499 CV06FC 21994930 IC50 = 3 nM T12499 CHN2Y3 21994942 IC50 = 100 nM T12499 C6DK9A 21994949 IC50 = 1330 nM T12499 CVA9P4 21994955 IC50 = 9 nM T12499 C1YF4W 21994961 IC50 = 9 nM T12499 C2BAM8 21994965 IC50 = 11 nM T12499 C8OBH7 21994981 IC50 = 6.2 nM T12499 CT17VP 21994984 IC50 = 240 nM T12499 C3C6FO 21994992 IC50 = 24 nM T12499 CA1CL8 21995003 IC50 = 26 nM T12499 CXJ26U 21995007 IC50 = 40 nM T12499 C12GPM 21995020 IC50 = 3170 nM T12499 CD7G2O 21995023 IC50 = 2.4 nM T12499 CEM56K 21995028 IC50 = 8 nM T12499 CP7R3X 21995029 IC50 = 18 nM T12499 CG35FE 21995041 IC50 = 3 nM T12499 CA16TP 21995049 IC50 = 4 nM T12499 C4NZJ6 21995088 IC50 = 50 nM T12499 CYR02Q 21995091 IC50 = 30 nM T12499 C7UQM9 21995099 IC50 > 12500 nM T12499 CXJI39 22022153 IC50 = 3000 nM T12499 CGX61W 22041319 IC50 = 65 nM T12499 CQ2XW6 22346679 IC50 = 74 nM T12499 CZRT79 22346947 IC50 = 50 nM T12499 C2AYF1 22634103 IC50 = 300 nM T12499 CZR4U0 22634116 IC50 = 90 nM T12499 CXP45U 22634145 IC50 = 80 nM T12499 C3CN7M 22634150 IC50 = 15 nM T12499 CUXV98 22634165 IC50 = 310 nM T12499 CMVL20 22634174 IC50 = 130 nM T12499 CCZ07D 22634175 IC50 = 700 nM T12499 C5E4BO 22634176 IC50 = 123 nM T12499 CT7MB6 22634192 IC50 = 55 nM T12499 C06DIG 22634197 IC50 = 565 nM T12499 CKX62Q 22634226 IC50 = 11 nM T12499 CWEL63 22634235 IC50 = 2010 nM T12499 C3CV5J 22634236 IC50 = 45 nM T12499 C5LXT1 22634281 IC50 = 337 nM T12499 C7H4DQ 22634288 IC50 = 100 nM T12499 CZE2U9 22634355 IC50 = 70 nM T12499 CEN7D5 22634359 IC50 = 7 nM T12499 CKOH73 22634360 IC50 = 1800 nM T12499 C68JBA 22634362 IC50 = 30 nM T12499 C54BIF 22634389 IC50 = 87 nM T12499 CH65IJ 22634393 IC50 = 1730 nM T12499 C6AE5O 22634424 IC50 = 330 nM T12499 C7OA9U 22634439 IC50 = 120 nM T12499 C7WX8F 22634450 IC50 = 39 nM T12499 C5P7OI 22634478 IC50 = 11 nM T12499 CAJ5E3 22634481 IC50 = 4 nM T12499 CD03MH 22634489 IC50 = 380 nM T12499 CI15AY 22634499 IC50 = 90 nM T12499 C1WRE8 22634507 IC50 = 7 nM T12499 CO4FX0 22634509 IC50 = 3120 nM T12499 CDQV06 22634522 IC50 = 19 nM T12499 CXSQ56 22634523 IC50 = 27 nM T12499 C4KY6D 22634526 IC50 > 12500 nM T12499 C5NP3B 22634530 IC50 = 85 nM T12499 C9P3CF 22634544 IC50 > 3125 nM T12499 CTWJ81 22634553 IC50 = 20 nM T12499 CNJ78C 22634560 IC50 = 15070 nM T12499 CSIO14 22634565 IC50 = 666 nM T12499 CLOR96 22736225 IC50 = 46 nM T12499 CT39NL 22736235 IC50 < 1 nM T12499 CAU62I 22736238 IC50 = 890 nM T12499 CV1OI5 22736332 IC50 = 42 nM T12499 C5ONK2 22736361 IC50 = 120 nM T12499 CT57UR 23075146 IC50 = 829000 nM T12499 CGV8M7 23375461 IC50 = 200 nM T12499 CG12OL 23518511 IC50 = 600 nM T12499 CE7K3W 23532567 IC50 > 10000 nM T12499 C5AZ7B 23536770 IC50 = 6 nM T12499 CW6OB1 23627212 IC50 = 260 nM T12499 CR3M1N 23644582 Ki = 20 nM T12499 C70VCY 23646368 IC50 = 20 nM T12499 CG6D4M 23647319 IC50 > 10000 nM T12499 CY8Z7X 23647330 IC50 > 10000 nM T12499 C4XD8H 23647348 IC50 > 10000 nM T12499 CI6C1R 23658582 IC50 = 75 nM T12499 CBXC05 24424330 IC50 = 31 nM T12499 C3RVK4 24750458 IC50 > 800 ug.mL-1 T12499 CA3I4T 24753787 IC50 > 50000 nM T12499 CHU49V 24757938 IC50 = 38 nM T12499 C7YG1N 24759534 IC50 = 19 nM T12499 CAJ4T2 24762205 IC50 = 22 nM T12499 CQNP54 24764449 IC50 = 1000 nM T12499 C2UOE0 24766030 IC50 = 46 nM T12499 C31EHS 24767187 IC50 > 100000 nM T12499 C4Z9CN 24769780 IC50 = 33 nM T12499 CJUK39 24770517 IC50 > 10000 nM T12499 CLBP72 24798571 IC50 = 4440 nM T12499 C9PA0M 24807809 IC50 > 30000 nM T12499 C0JUN4 24812717 IC50 = 19 nM T12499 CP6N9M 24812718 IC50 = 1900 nM T12499 CW0G8H 24812719 IC50 = 1700 nM T12499 CO9Z0H 24822598 IC50 = 1100 nM T12499 C51IZL 24822599 IC50 = 1300 nM T12499 CA90EF 24822600 IC50 = 1800 nM T12499 CCP2M3 24822704 IC50 > 50000 nM T12499 C4A6LB 24823090 IC50 = 2000 nM T12499 C2B4JP 24823091 IC50 = 4300 nM T12499 C14FLQ 24823250 IC50 = 25000 nM T12499 C3KPO7 24823251 IC50 = 1000 nM T12499 C3A2BF 24823416 IC50 = 4600 nM T12499 CYBI02 24823426 IC50 = 15 nM T12499 C45UGH 24823586 IC50 = 0.5 nM T12499 CFA3T8 24823588 IC50 = 14 nM T12499 C51ZTV 24823589 IC50 = 5 nM T12499 CX0QC1 24823590 IC50 = 0.8 nM T12499 CR7CH6 24823736 IC50 = 10 nM T12499 C26KXV 24823738 IC50 = 6 nM T12499 CO3K7R 24823740 IC50 = 1.8 nM T12499 CBLJ48 24823898 IC50 = 6 nM T12499 CG0K1Z 24824046 IC50 = 239 nM T12499 CDT3L2 24824050 IC50 = 27 nM T12499 CLN48F 24824051 IC50 = 90 nM T12499 C0NXE2 24824052 IC50 = 1500 nM T12499 CWTI12 24824188 IC50 = 500 nM T12499 CQ1A8W 24824189 IC50 = 19 nM T12499 C8RE5C 24824190 IC50 > 4000 nM T12499 C3K1FM 24824191 IC50 > 4000 nM T12499 CV0S5L 24824318 IC50 = 2200 nM T12499 CUK14T 24824319 IC50 > 4000 nM T12499 CZ09ID 24824320 IC50 = 2400 nM T12499 CM28KX 24824321 IC50 = 1000 nM T12499 CD57UN 24824322 IC50 = 150 nM T12499 CNI50G 24824323 IC50 = 78 nM T12499 C84VZK 24824448 IC50 = 1000 nM T12499 C6OC4K 24824449 IC50 = 1300 nM T12499 C5BA7V 24824452 IC50 = 21 nM T12499 CR49SP 24824453 IC50 > 4000 nM T12499 CG64EL 24824454 IC50 > 4000 nM T12499 CM28WD 24825721 IC50 > 10000 nM T12499 CX0S9L 24854902 IC50 = 6048 nM T12499 C1SVT2 24854903 IC50 > 5000 nM T12499 C61KPI 24856363 IC50 > 16000 nM T12499 CS82HN 24856408 IC50 = 37 nM T12499 CZ5Y4H 24856498 IC50 = 23 nM T12499 CC10FW 24857629 IC50 = 92 nM T12499 CCS58O 24863072 IC50 = 21 nM T12499 C6C2GX 24863500 IC50 = 23 nM T12499 CYVB83 24863584 IC50 = 210 nM T12499 CQ15ML 24863670 IC50 = 78 nM T12499 C4XZ3N 24863671 IC50 = 110 nM T12499 CSW5V3 24865437 IC50 = 24000 nM T12499 CE3IW4 24879184 IC50 = 340 nM T12499 C7V8BA 24879242 IC50 = 480 nM T12499 CT76XV 24879243 IC50 = 740 nM T12499 CGD8J5 24879244 IC50 = 230 nM T12499 C1XWO7 24879245 IC50 = 110 nM T12499 CA21RX 24879305 IC50 = 580 nM T12499 COF05N 24879306 IC50 = 1700 nM T12499 C6NIQ2 24879307 IC50 = 7.2 nM T12499 C45HIT 24879308 IC50 = 1200 nM T12499 CM6G7A 24879309 IC50 = 150 nM T12499 C0KW5Y 24879310 IC50 = 410 nM T12499 C7M9FB 24879311 IC50 = 25000 nM T12499 C0ZJX6 24879366 IC50 = 570 nM T12499 C5NA4Z 24879367 IC50 = 1800 nM T12499 CDJE41 24879368 IC50 = 7800 nM T12499 C4MG3B 24882476 IC50 = 0.6 nM T12499 C43HWQ 24883287 IC50 = 300 nM T12499 C8DA5Q 24883334 IC50 < 100 nM T12499 C0P6AU 24894017 IC50 < 1 nM T12499 CY8L7E 24896769 IC50 > 10000 nM T12499 C5ZM4T 24936119 IC50 = 7 nM T12499 C8DG1Y 24941253 IC50 > 10000 nM T12499 CLZ23U 24951610 IC50 > 30000 nM T12499 CU7I2E 24963046 IC50 = 122 nM T12499 CD5HQ0 24969301 IC50 > 10000 nM T12499 CT8OF0 24983254 IC50 = 25 nM T12499 CVF62Q 24983255 IC50 = 80 nM T12499 CX6FR3 24983298 IC50 = 4799 nM T12499 CEQ1F2 24983299 IC50 = 269 nM T12499 CQ46VT 24983495 IC50 = 292 nM T12499 C4EG8R 24993189 IC50 > 10000 nM T12499 CS3Q8B 24995659 IC50 > 2000 nM T12499 C6P1CX 25066843 IC50 = 28 nM T12499 C2KY1G 25094210 IC50 = 468 nM T12499 CTG49K 25110690 IC50 = 14 nM T12499 CG3XC9 25124150 IC50 = 1200 nM T12499 CO2IR5 25124816 IC50 > 3000 nM T12499 CF7C5B 25129829 IC50 > 10000 nM T12499 CXNM84 25129830 IC50 = 3814 nM T12499 CY2S1P 25129831 IC50 > 10000 nM T12499 C36FXD 25138012 IC50 = 14 nM T12499 CQMU82 25138148 IC50 = 0.4 nM T12499 CD9O6K 25138149 IC50 = 7 nM T12499 CO6N7P 25138154 IC50 > 25000 nM T12499 CGT1W6 25144294 IC50 = 12 nM T12499 CU7VR0 25144732 IC50 <= 1 nM T12499 C65YQG 25145144 IC50 = 384 nM T12499 C6BWZ8 25145145 IC50 = 2353 nM T12499 C78YWA 25145716 IC50 = 271 nM T12499 CL47VI 25145718 IC50 = 45 nM T12499 CSO82D 25154877 Ki = 0.04 nM T12499 CR0S2O 25195244 IC50 = 6 nM T12499 CNG96H 25210579 IC50 > 10000 nM T12499 CNQ9G5 25218180 IC50 < 1000 nM T12499 CRO8T9 25263033 Ki = 11 nM T12499 CC71QJ 27666048 IC50 = 10900 nM T12499 CXG02H 42226845 IC50 = 10000 nM T12499 CWS37O 42618140 IC50 > 25118.86 nM T12499 C2JV3O 42618143 IC50 = 15848.93 nM T12499 CG01BO 42618144 IC50 = 19952.62 nM T12499 CI9DK5 42628614 IC50 = 1300 nM T12499 CU9E4P 42629114 IC50 > 10000 nM T12499 CO42DC 44138048 IC50 > 10000 nM T12499 CL65QV 44138049 IC50 > 10000 nM T12499 CLW80F 44160269 IC50 = 2900 nM T12499 CO6HU7 44178069 IC50 = 731 nM T12499 CCFQ29 44187005 IC50 = 505 nM T12499 CEL61X 44229839 IC50 = 1700 nM T12499 CG1C9E 44269392 IC50 > 250000 nM T12499 CAT6W7 44269404 IC50 > 250000 nM T12499 C4SA3Y 44269518 IC50 > 250000 nM T12499 CVE17U 44271480 IC50 = 22000 nM T12499 CMZD96 44276805 IC50 > 2000 nM T12499 CDM14R 44277152 IC50 = 7.4 nM T12499 CFKY97 44277389 IC50 = 170 nM T12499 CP4Z9O 44277406 IC50 = 7700 nM T12499 C7AMH2 44277415 IC50 = 2800 nM T12499 CDSK68 44277416 IC50 = 30 nM T12499 CX0R6Z 44277458 IC50 = 400 nM T12499 CT03HW 44277459 IC50 = 17000 nM T12499 CP3FK1 44277464 IC50 > 12500 nM T12499 C6ILO7 44277479 IC50 = 1900 nM T12499 C54EAR 44277500 IC50 = 350000 nM T12499 CY9S4U 44277503 IC50 = 10000 nM T12499 CTOR69 44277507 IC50 = 1100 nM T12499 CM4QB2 44277523 IC50 = 1600 nM T12499 CTUE56 44277530 IC50 = 810 nM T12499 C94XTC 44277552 IC50 = 1900 nM T12499 C25XAV 44277553 IC50 = 6000 nM T12499 CM8ZU1 44277554 IC50 = 8500 nM T12499 CH70ZJ 44277555 IC50 = 2000 nM T12499 CT2C8Y 44277556 IC50 = 100 nM T12499 C7GVH2 44277568 IC50 = 1600 nM T12499 C0R5LM 44277575 IC50 = 1200 nM T12499 C48NAJ 44277576 IC50 = 1100 nM T12499 CC09ZV 44277619 IC50 = 1800 nM T12499 CF39VK 44277620 IC50 = 1200 nM T12499 CN26TB 44277621 IC50 = 1800 nM T12499 CUCN89 44277736 IC50 = 10 nM T12499 CHOA91 44277745 IC50 = 69 nM T12499 CNZR96 44277759 IC50 = 238 nM T12499 CQ2Y5R 44277762 IC50 = 53 nM T12499 CZ9NX1 44277837 IC50 = 60 nM T12499 COPF86 44277899 IC50 = 1600 nM T12499 CA74WK 44277900 IC50 = 1500 nM T12499 C6EJ0W 44278090 IC50 = 665 nM T12499 CG84EI 44278256 IC50 = 6.2 nM T12499 CZFQ76 44291533 IC50 = 19 nM T12499 CTX6L9 44293106 IC50 = 242000 nM T12499 CZ8W0T 44293432 IC50 > 2094000 nM T12499 CH3J2E 44299176 IC50 = 80 nM T12499 C27GVO 44299203 IC50 = 800 nM T12499 CY6WC0 44299236 IC50 = 400 nM T12499 C3RG0C 44299304 IC50 = 700 nM T12499 CJM26I 44299321 IC50 = 300 nM T12499 C9UGL3 44299325 IC50 = 700 nM T12499 CJEZ96 44299338 IC50 = 500 nM T12499 CNH34G 44299354 IC50 = 400 nM T12499 C82MSD 44299360 IC50 = 700 nM T12499 CF1N4E 44307877 IC50 = 178000 nM T12499 CD9J2B 44308029 IC50 = 638000 nM T12499 CC07XF 44308301 IC50 > 12500 nM T12499 CPK13M 44308362 IC50 = 110 nM T12499 C5P1AZ 44308363 IC50 > 12500 nM T12499 C5KA1C 44308378 IC50 > 12500 nM T12499 CM3O2B 44308391 IC50 = 3230 nM T12499 CWJ3T4 44308408 IC50 = 7250 nM T12499 C2X3TN 44308485 IC50 = 4400 nM T12499 CG8U6C 44308486 IC50 = 200 nM T12499 CG47MH 44308503 IC50 > 12500 nM T12499 C0M1IY 44308504 IC50 > 12500 nM T12499 C6PEF5 44308506 IC50 > 12500 nM T12499 C0XY4O 44308544 IC50 = 272 nM T12499 CP76DF 44308560 IC50 > 12500 nM T12499 C1S6MR 44308561 IC50 = 5600 nM T12499 C8MN4Y 44308567 IC50 > 12500 nM T12499 CB85WM 44308568 IC50 = 90 nM T12499 CMZI25 44308570 IC50 = 70 nM T12499 C13DBO 44308571 IC50 > 12500 nM T12499 C46QFM 44308664 IC50 > 12500 nM T12499 C2ZJH7 44308683 IC50 > 12500 nM T12499 CE5T3I 44308684 IC50 = 23000 nM T12499 CS1W5Z 44308685 IC50 > 12500 nM T12499 CEU2W4 44308690 IC50 < 2 nM T12499 C8EVZ0 44308700 IC50 > 12500 nM T12499 CWY9N5 44308701 IC50 = 4270 nM T12499 CIYE50 44308712 IC50 > 12500 nM T12499 C4U1MP 44308728 IC50 > 12500 nM T12499 CPA69W 44308729 IC50 = 3 nM T12499 CY6ZB5 44308830 IC50 = 220 nM T12499 C1I6RG 44308968 IC50 < 3 nM T12499 C1I0LN 44308993 IC50 < 3 nM T12499 CKVZ38 44308994 IC50 = 40 nM T12499 CF9I2S 44309110 IC50 = 1490 nM T12499 C8VX1L 44309229 IC50 = 942 nM T12499 CZQ4S0 44309230 IC50 < 3 nM T12499 CHF28G 44309494 IC50 = 131 nM T12499 CE9Z6L 44319231 IC50 = 820 nM T12499 CRWF80 44319232 IC50 = 2680 nM T12499 CF3QW5 44319234 IC50 = 3170 nM T12499 CFQ2L8 44319256 IC50 = 3170 nM T12499 CEL1H2 44319376 IC50 = 24 nM T12499 C4M6VJ 44319377 IC50 = 26 nM T12499 C7PS2Z 44319406 IC50 = 9 nM T12499 C9AT6W 44319420 IC50 = 4 nM T12499 C61ISW 44319421 IC50 = 2 nM T12499 CE1XR0 44319422 IC50 = 5 nM T12499 C6A0ZG 44319438 IC50 = 7 nM T12499 CIK71G 44319439 IC50 = 10 nM T12499 C3DXJ2 44319445 IC50 = 3 nM T12499 CIP4B3 44319451 IC50 = 9.4 nM T12499 CW5AR2 44319455 IC50 = 21 nM T12499 CUC1O5 44319479 IC50 = 4 nM T12499 CTKI85 44319593 IC50 = 100 nM T12499 C3Y4AS 44319618 IC50 = 15 nM T12499 CY5WL6 44319619 IC50 = 70 nM T12499 CKN3C5 44319631 IC50 = 26 nM T12499 C8ZF6H 44320538 IC50 > 3100 nM T12499 C4KS5N 44320732 IC50 = 1.1 nM T12499 CI6W3R 44320738 IC50 = 6 nM T12499 CC6YI7 44320769 Ki = 0.54 nM T12499 CBN1H4 44320801 IC50 = 403 nM T12499 C2USC1 44320802 IC50 > 3100 nM T12499 CTI86J 44320812 IC50 = 1890 nM T12499 C38YXS 44320815 IC50 = 2 nM T12499 C16ATL 44320820 IC50 > 3100 nM T12499 C6XRM9 44320821 IC50 = 1740 nM T12499 CMJ4Y2 44320829 IC50 = 1 nM T12499 CN7MI0 44320840 IC50 > 3100 nM T12499 CIQ1Y8 44320841 IC50 > 3100 nM T12499 C0WNK8 44320856 IC50 > 3100 nM T12499 C2C3HQ 44320857 IC50 > 3100 nM T12499 CL86PD 44320858 IC50 > 3100 nM T12499 C5WA0P 44320868 IC50 = 13 nM T12499 C9E2WN 44320869 IC50 = 10 nM T12499 C2B9QV 44320870 IC50 = 138 nM T12499 CKHP01 44320871 IC50 = 180 nM T12499 CCBU40 44320872 IC50 = 72 nM T12499 CP64WV 44320885 IC50 = 32 nM T12499 CJZ26I 44320905 IC50 = 8 nM T12499 C5JBP7 44320912 IC50 = 6 nM T12499 CE4OA6 44320964 IC50 > 3100 nM T12499 CR8Q1U 44320965 IC50 = 15 nM T12499 CK2X4T 44321004 IC50 = 5 nM T12499 CTJ69K 44321005 IC50 = 8 nM T12499 CD72YE 44321008 IC50 = 27 nM T12499 C29TOE 44321009 IC50 = 84 nM T12499 CI9U1O 44321055 IC50 = 20 nM T12499 CO0E8Y 44321057 IC50 = 17 nM T12499 CC68EY 44321060 IC50 = 1590 nM T12499 CBZ15Y 44321061 IC50 = 9 nM T12499 C14SKY 44321062 IC50 = 9 nM T12499 CO6T2M 44321063 IC50 = 403 nM T12499 CMX7N1 44321092 IC50 = 31 nM T12499 C7RE2Q 44321105 IC50 = 20 nM T12499 C3V4CY 44321106 IC50 = 5 nM T12499 CGNQ90 44321109 IC50 = 35 nM T12499 C1UE2V 44321110 IC50 = 13 nM T12499 CL6TY5 44321118 IC50 = 77 nM T12499 C9UTH8 44321136 IC50 = 21 nM T12499 CJ4Q9Z 44321140 IC50 = 20 nM T12499 C6OJ7A 44321151 IC50 = 3 nM T12499 C5TNF7 44321155 IC50 = 53 nM T12499 CLV2C0 44321167 IC50 = 7 nM T12499 C1LFI2 44321182 IC50 = 6 nM T12499 C74NLZ 44321198 IC50 = 10 nM T12499 C0PX6H 44321252 IC50 = 2 nM T12499 C3XB0U 44321258 IC50 = 6 nM T12499 C82NIY 44321259 IC50 = 8 nM T12499 CXM61A 44321260 IC50 = 2 nM T12499 CLAS90 44321316 IC50 = 235 nM T12499 CQX6F9 44321339 IC50 > 3100 nM T12499 CFD31S 44321340 IC50 = 327 nM T12499 C2Y3NE 44321361 IC50 = 1 nM T12499 C2FST3 44324647 IC50 = 81 nM T12499 CI8YR0 44324649 IC50 = 3800 nM T12499 C7JYP4 44324728 IC50 = 27000 nM T12499 CY69SU 44324769 IC50 = 18000 nM T12499 C3PED0 44331665 IC50 = 36000 nM T12499 CLG7Q6 44337120 IC50 = 6 nM T12499 CCGB45 44337122 IC50 = 2 nM T12499 CVW4D1 44337132 IC50 = 10 nM T12499 CE2AV7 44337155 IC50 = 5 nM T12499 CW4Q0X 44337161 IC50 = 7 nM T12499 CLB03R 44337267 IC50 = 3 nM T12499 C3LO9F 44337272 IC50 = 26 nM T12499 CC3BV7 44337290 IC50 = 7 nM T12499 CG7I6O 44337337 IC50 = 10 nM T12499 C7S6FQ 44337369 IC50 = 70 nM T12499 CQ2W7M 44337378 IC50 = 9 nM T12499 CP64NY 44337501 IC50 = 5 nM T12499 CSC40Y 44337509 IC50 = 5.4 nM T12499 CVP9L5 44337524 IC50 = 10 nM T12499 CH26ZA 44343296 IC50 > 10000 nM T12499 C2OMC0 44343708 IC50 > 500000 nM T12499 CQZM34 44355143 IC50 > 100000 nM T12499 CX1I0D 44355168 IC50 > 50000 nM T12499 C2F9DZ 44355323 IC50 > 100000 nM T12499 C4LKS3 44355443 IC50 = 10000 nM T12499 CJWK61 44355456 IC50 > 50000 nM T12499 C9YI1R 44355486 IC50 = 2500 nM T12499 CO5S7X 44379379 IC50 > 2000000 nM T12499 C6LSB4 44381409 IC50 = 340 nM T12499 C6LC8M 44381556 IC50 = 620 nM T12499 CC35RY 44386906 IC50 = 9650 nM T12499 C7PBJ8 44405918 IC50 = 2350 nM T12499 C0GR5F 44405919 IC50 = 3480 nM T12499 CO5WU8 44405977 IC50 = 8960 nM T12499 C9LX5Q 44406001 IC50 = 23200 nM T12499 CQ4U7T 44406037 IC50 = 106 nM T12499 CEVF48 44406058 IC50 = 9180 nM T12499 CF46WP 44406078 IC50 = 318 nM T12499 CUQ6R8 44406079 IC50 = 54 nM T12499 CG2W4V 44406138 IC50 > 50000 nM T12499 CV09DY 44410717 IC50 > 10000 nM T12499 CP3CI1 44410720 IC50 > 10000 nM T12499 C8W7AD 44410723 IC50 > 10000 nM T12499 CAT5X4 44410829 IC50 > 10000 nM T12499 CC6Y5P 44410844 IC50 > 10000 nM T12499 CG34TY 44410851 IC50 > 10000 nM T12499 C41EIA 44410869 IC50 > 10000 nM T12499 CB6AE8 44410948 IC50 > 10000 nM T12499 CXZG12 44410949 IC50 > 10000 nM T12499 CS7IE9 44410953 IC50 > 10000 nM T12499 CA9M4X 44410954 IC50 > 10000 nM T12499 C3SP5H 44410955 IC50 > 10000 nM T12499 C5D6YP 44410956 IC50 > 10000 nM T12499 C5W1VC 44410959 IC50 > 10000 nM T12499 CM1C2G 44410960 IC50 > 10000 nM T12499 CVSI80 44411048 IC50 > 10000 nM T12499 CN72BR 44411161 IC50 > 10000 nM T12499 C4AW0O 44411183 IC50 > 10000 nM T12499 C0WQ2A 44412535 IC50 > 10000 nM T12499 C9EL3N 44412536 IC50 > 10000 nM T12499 CCP34J 44412547 IC50 = 971 nM T12499 C0JW3X 44412548 IC50 = 2350 nM T12499 C71GSY 44412549 IC50 > 10000 nM T12499 C8YIO7 44412564 IC50 = 229 nM T12499 CD0XK4 44412565 IC50 = 1450 nM T12499 C45MBP 44412566 IC50 = 5990 nM T12499 C2Z9QT 44412568 IC50 = 32 nM T12499 CUAQ42 44412569 IC50 = 149 nM T12499 CIF8K3 44412570 IC50 = 52 nM T12499 C6IUQ8 44412571 IC50 = 3 nM T12499 C7C2NQ 44412577 IC50 = 708 nM T12499 CRHK90 44412586 IC50 = 28 nM T12499 C8WX2G 44412587 IC50 = 96 nM T12499 CRA02Z 44412602 IC50 = 418 nM T12499 C42YIW 44412603 IC50 > 10000 nM T12499 CR18DN 44412728 IC50 = 4 nM T12499 C7LBS4 44412754 IC50 > 10000 nM T12499 C6P9LY 44412768 IC50 > 10000 nM T12499 C4KR2P 44412769 IC50 = 2580 nM T12499 CSL1C7 44412787 IC50 > 10000 nM T12499 CV12PJ 44412788 IC50 = 155 nM T12499 CO0R3U 44412789 IC50 = 3 nM T12499 CT1EU9 44412790 IC50 = 4 nM T12499 C5JQ0S 44412804 IC50 > 10000 nM T12499 CZE9H2 44412805 IC50 = 4490 nM T12499 C1XOC5 44412806 IC50 = 230 nM T12499 CFB16V 44412829 IC50 = 1820 nM T12499 CA6GK9 44412842 IC50 = 3130 nM T12499 CLS5H6 44412843 IC50 = 301 nM T12499 CP9KT1 44412856 IC50 = 190 nM T12499 CNJS19 44412857 IC50 = 4290 nM T12499 CS05HP 44412870 IC50 = 6 nM T12499 C50CHI 44412871 IC50 = 9 nM T12499 C4TD2F 44412992 IC50 = 3860 nM T12499 C0F3NI 44414305 IC50 = 143 nM T12499 C6FY3V 44414306 IC50 = 26 nM T12499 C3E4AR 44414321 IC50 = 43 nM T12499 C7KZV2 44414322 IC50 = 21141 nM T12499 CJM06T 44414347 IC50 > 50000 nM T12499 C8R4PT 44414468 IC50 = 182 nM T12499 CXR08Z 44414469 IC50 = 2814 nM T12499 CE1V5J 44414487 IC50 = 71 nM T12499 CBSJ78 44414580 IC50 = 21 nM T12499 C3Z7VW 44414581 IC50 = 3 nM T12499 CC8R6T 44414609 IC50 = 4802 nM T12499 CRB78V 44414623 IC50 = 2837 nM T12499 C8ED2X 44414624 IC50 = 10 nM T12499 CXTJ75 44414636 IC50 = 179 nM T12499 CH0VO6 44414656 IC50 = 7269 nM T12499 CCF69N 44414657 IC50 = 285 nM T12499 C8G5YN 44415111 IC50 = 1 nM T12499 CHJ7T1 44415158 IC50 = 1 nM T12499 C5TQ4F 44415291 IC50 = 1 nM T12499 C32UJZ 44419930 IC50 = 7700 nM T12499 CR2WY4 44419931 IC50 > 10000 nM T12499 C9Y1FS 44419937 IC50 > 10000 nM T12499 CAP2D3 44419938 IC50 = 1286 nM T12499 C2I3LY 44419942 IC50 = 294 nM T12499 CC31RB 44419943 IC50 = 79 nM T12499 CCV9U5 44419947 IC50 = 384 nM T12499 CXUV94 44419948 IC50 = 71 nM T12499 C76LAG 44419953 IC50 = 137 nM T12499 C3C0SW 44419954 IC50 = 3 nM T12499 CSFI82 44419961 IC50 = 17 nM T12499 CB47IS 44419962 IC50 = 65 nM T12499 C6W7YQ 44419967 IC50 = 44 nM T12499 CX1U0E 44419972 IC50 = 130 nM T12499 CSH8I0 44419973 IC50 = 45 nM T12499 CS83YT 44419977 IC50 = 165 nM T12499 C2SZ3E 44419978 IC50 = 519 nM T12499 CL4O8E 44419981 IC50 = 43 nM T12499 C25NUJ 44419988 IC50 = 333 nM T12499 CA9K5Y 44419989 IC50 = 193 nM T12499 CKWI23 44419990 IC50 > 10000 nM T12499 CTC09S 44419991 IC50 = 4.2 nM T12499 CK93IX 44419994 IC50 = 5564 nM T12499 C3N6EX 44419995 IC50 = 8640 nM T12499 CCS6L8 44419998 IC50 > 10000 nM T12499 C9RBH4 44419999 IC50 = 24 nM T12499 C26YUL 44420000 IC50 = 6.8 nM T12499 C8HOG7 44422489 IC50 = 20 nM T12499 CBS5K2 44432304 IC50 = 17600 nM T12499 CFJX63 44432305 IC50 = 240 nM T12499 C54URN 44432306 IC50 = 541 nM T12499 C57FJN 44432307 IC50 = 130 nM T12499 C0PHT6 44432309 IC50 = 4470 nM T12499 CA9SP2 44432315 IC50 = 31 nM T12499 CL05KJ 44438314 IC50 = 1210 nM T12499 C3XQK1 44438318 IC50 = 6 nM T12499 CSB51N 44438320 IC50 = 6 nM T12499 CGV37F 44440254 IC50 = 16038 nM T12499 C5JUV3 44440256 IC50 > 50000 nM T12499 CFB56S 44440259 IC50 = 21382 nM T12499 CEW9G2 44440261 IC50 = 26529 nM T12499 CI9W8E 44447914 IC50 = 3310 nM T12499 CUB12D 44449577 IC50 = 185 nM T12499 CDV6X9 44454507 IC50 = 7 nM T12499 C6SMY7 44454538 IC50 = 53 nM T12499 CZI92T 44454651 IC50 = 84 nM T12499 CIA39D 44454676 IC50 = 45 nM T12499 C7DGA2 44454678 IC50 = 19 nM T12499 C1F3LT 44454702 IC50 = 22 nM T12499 CCW57R 44454703 IC50 = 101 nM T12499 CFS7W2 44454728 IC50 = 25 nM T12499 CTL43P 44454729 IC50 = 41 nM T12499 CZC95J 44454731 IC50 = 44 nM T12499 CIB24G 44457163 IC50 > 12500 nM T12499 CN8HV0 44457164 IC50 = 60 nM T12499 C3I6ZY 44457241 IC50 = 810 nM T12499 C67VXQ 44457503 IC50 = 1 nM T12499 C71EPS 44460198 IC50 = 7.5 ug.mL-1 T12499 C3PAD4 44460222 IC50 > 10 ug.mL-1 T12499 CLNZ91 44460237 IC50 > 10 ug.mL-1 T12499 C9Z8XJ 44460238 IC50 = 1.2 ug.mL-1 T12499 CH9F0N 44460247 IC50 > 10 ug.mL-1 T12499 CV1Q0D 44460258 IC50 = 0.62 ug.mL-1 T12499 CF9Z3W 44461749 IC50 = 710 nM T12499 C84RLC 44461768 IC50 = 1500 nM T12499 C3WV2D 44461769 IC50 = 310 nM T12499 C5KD6H 44461778 IC50 = 5000 nM T12499 CGR15K 44461807 IC50 = 1400 nM T12499 CW5QX9 44461811 IC50 = 470 nM T12499 COK3T6 44461852 IC50 = 1700 nM T12499 CN0P6M 44461863 IC50 = 5000 nM T12499 CNW9M3 44461865 IC50 = 110 nM T12499 CEDL98 44461873 IC50 = 880 nM T12499 CXDB59 44461880 IC50 = 600 nM T12499 C24SNH 44461881 IC50 > 5000 nM T12499 CFJ28C 44461889 IC50 = 1000 nM T12499 CH7M6G 44461919 IC50 = 1700 nM T12499 CF08CB 44462184 IC50 > 5000 nM T12499 CJ3QZ6 44462200 IC50 = 32 nM T12499 CQ3PB5 44462201 IC50 = 5000 nM T12499 C5WL1F 44473009 IC50 = 1200 nM T12499 CEG1S5 44473011 IC50 = 600 nM T12499 C46OMR 44473016 IC50 = 47000 nM T12499 C7N2AQ 44473101 IC50 = 280 nM T12499 C4MG3F 44473102 IC50 = 12 nM T12499 CA85NJ 44473103 IC50 = 150 nM T12499 CYH6P3 44520205 IC50 = 566 nM T12499 CWPT02 44555415 IC50 = 0.12 nM T12499 C3VRO9 44557921 IC50 > 10000 nM T12499 CF16QB 44560451 IC50 = 546 nM T12499 C0U8DH 44560546 IC50 = 2760 nM T12499 C3XTA7 44562721 Ki = 13 nM T12499 CO3SK5 44563262 IC50 = 220 nM T12499 C3HW7L 44570553 IC50 > 30000 nM T12499 C17PVE 44570554 IC50 > 30000 nM T12499 CLOY92 44570599 IC50 = 500 nM T12499 CK06LT 44570600 IC50 = 7000 nM T12499 CJY8S0 44570884 IC50 = 38000 nM T12499 CWFB42 44571820 IC50 = 710 nM T12499 CW8P9Y 44576189 IC50 = 7000 nM T12499 C9VXN3 44578709 IC50 > 10000 nM T12499 C3J9AT 44578884 IC50 = 1167 nM T12499 CA7R2X 44579356 EC50 = 14400 nM T12499 CNS6A4 44579357 EC50 = 23300 nM T12499 C31TFG 44579358 EC50 = 18400 nM T12499 C53ZVU 44579359 IC50 = 50000 nM T12499 CM9TC5 44579360 EC50 > 150000 nM T12499 CV01SB 44579361 EC50 = 4400 nM T12499 C7Q1VU 44580077 IC50 = 6000 nM T12499 CL90SE 44580358 IC50 = 2000 nM T12499 CK1VE7 44580420 IC50 = 8000 nM T12499 CH2R7X 44580449 IC50 = 3000 nM T12499 C1VH0C 44580532 IC50 > 16000 nM T12499 CXC52J 44580649 IC50 = 3000 nM T12499 CE32BQ 44580689 IC50 = 70 nM T12499 C8Z5AX 44580778 IC50 = 1000 nM T12499 C6RJZ5 44581565 IC50 = 48 nM T12499 CV5GD1 44589002 IC50 = 180 nM T12499 C83KEG 44589022 IC50 = 590 nM T12499 CL3DO5 44593603 IC50 = 100 ug.mL-1 T12499 C4EP8N 44593604 IC50 > 800 ug.mL-1 T12499 C3KS6C 44593605 IC50 = 700 ug.mL-1 T12499 C8WX5D 44593606 IC50 > 800 ug.mL-1 T12499 CU3RF1 45139989 IC50 > 10000 nM T12499 CQGZ06 45139991 IC50 > 10000 nM T12499 C6F8UE 45261965 IC50 = 10000 nM T12499 C0T2MQ 45262036 IC50 = 20000 nM T12499 CKQ5U9 45266326 IC50 > 1936000 nM T12499 C5Q4DT 45266328 IC50 > 2088000 nM T12499 COE8U0 45267045 IC50 = 41000 nM T12499 CY83PR 45267327 IC50 = 300 nM T12499 C84QFJ 45269074 IC50 > 1000 nM T12499 C3DH8I 45273358 IC50 > 1000 nM T12499 C6E2SC 45482700 IC50 > 10000 nM T12499 CZXH74 45482750 IC50 > 10000 nM T12499 C5S8MA 45485083 IC50 = 520 nM T12499 CZ8GR7 45486752 IC50 = 2073 nM T12499 C0D5TG 45486762 IC50 = 1770 nM T12499 CD40LR 45486763 IC50 = 1.5 nM T12499 C2D7YJ 45486771 IC50 = 47 nM T12499 CH4VY9 45486772 IC50 = 243 nM T12499 CP5YK9 45486775 IC50 = 0.06 nM T12499 CPC7I2 45486776 IC50 = 0.07 nM T12499 CG7RM9 45486777 IC50 = 1 nM T12499 CNC7M3 45486780 IC50 = 106 nM T12499 CZN60P 45486785 IC50 = 203 nM T12499 C1BMI3 45486789 IC50 > 1000 nM T12499 CPJD02 45486792 IC50 = 0.4 nM T12499 CB49PG 45486793 IC50 = 0.07 nM T12499 CR41JA 45486794 IC50 = 0.2 nM T12499 C4NTY8 45486795 IC50 = 1.8 nM T12499 CT4IR9 45486796 IC50 = 0.2 nM T12499 CXC03L 45486797 IC50 = 0.45 nM T12499 C3W9RC 45486798 IC50 = 115 nM T12499 CSK69U 45486806 IC50 > 20000 nM T12499 CTU89Y 45486814 IC50 = 110 nM T12499 CW2Q6T 45486815 IC50 = 10 nM T12499 CW42YX 45487634 IC50 > 1000 nM T12499 CG92CF 46175112 IC50 = 9200 nM T12499 C96BNW 46179972 IC50 = 35 nM T12499 CZBL95 46220496 IC50 = 18 nM T12499 CY3HW5 46224684 IC50 = 4600 nM T12499 C2P9QO 46228508 IC50 = 584 nM T12499 C6E5PY 46228822 IC50 > 10000 nM T12499 C3T8AM 46228951 IC50 = 5020 nM T12499 CYT37A 46232443 IC50 > 50000 nM T12499 C48ZVW 46232555 IC50 = 14000 nM T12499 CS9B1U 46232556 IC50 = 28000 nM T12499 C7ON5A 46233287 IC50 > 10000 nM T12499 CQW97N 46846072 IC50 = 790 nM T12499 COTJ39 46863083 IC50 = 1000 nM T12499 C7H4YM 46865419 IC50 > 10000 nM T12499 CC2O9R 46865656 IC50 = 5011.87 nM T12499 CX43UQ 46871756 IC50 = 7 nM T12499 CLS29B 46872626 IC50 > 10000 nM T12499 CRS61F 46879438 IC50 = 702 nM T12499 C27JEF 46879439 IC50 = 22 nM T12499 CF0T8P 46879440 IC50 = 406 nM T12499 C12RMW 46879441 IC50 = 38 nM T12499 CH2D7N 46879442 IC50 = 19 nM T12499 CI6OD8 46879443 IC50 = 38 nM T12499 C7YD4Q 46879444 IC50 = 11 nM T12499 C8MN5Q 46879445 IC50 = 18 nM T12499 CX6SW2 46879446 IC50 = 275 nM T12499 CNF3V6 46879447 IC50 = 4456 nM T12499 CW46VY 46879448 IC50 = 12 nM T12499 CLK6X3 46879907 IC50 = 58 nM T12499 CRPU47 46879908 IC50 = 7 nM T12499 C1TIE9 46880013 IC50 = 715 nM T12499 C2A8KO 46880066 IC50 = 230 nM T12499 CBRP80 46880067 IC50 = 23 nM T12499 C3FY2B 46880068 IC50 = 13 nM T12499 CX89TY 46880069 IC50 = 5 nM T12499 CB0XY1 46880070 IC50 = 26 nM T12499 CUD81V 46880071 IC50 = 38 nM T12499 CZP58Q 46880072 IC50 = 71 nM T12499 CC8OF9 46880073 IC50 = 204 nM T12499 CF41HG 46880098 IC50 = 132 nM T12499 C6O2YG 46880099 IC50 = 83 nM T12499 CI78DM 46880100 IC50 = 7 nM T12499 CU04ZK 46880101 IC50 = 16 nM T12499 C4E0MF 46880133 IC50 = 17 nM T12499 COJ16A 46880134 IC50 = 43 nM T12499 C71MGJ 46880135 IC50 = 63 nM T12499 C3R6TL 46880213 IC50 = 90 nM T12499 CT8BQ4 46880214 IC50 = 2280 nM T12499 C0JTO4 46880215 IC50 = 616 nM T12499 CAFN49 46880216 IC50 > 2500 nM T12499 CMVZ46 46886319 Ki = 39.81 nM T12499 C2O8RZ 46886323 IC50 = 71 nM T12499 CM02UJ 46890253 IC50 = 387 nM T12499 CB7VI8 46890254 IC50 = 10000 nM T12499 C7V3IA 46890314 IC50 = 4087 nM T12499 CHE6A1 46890315 IC50 = 1856 nM T12499 C1YS5A 46890918 IC50 = 28 nM T12499 CJ5S3N 46890968 IC50 = 4 nM T12499 CAGE32 46890969 IC50 = 23 nM T12499 C3A7BP 46890970 IC50 = 24 nM T12499 CTV73J 46890971 IC50 = 16 nM T12499 CUX9B4 46891024 IC50 = 8 nM T12499 CG35WP 46891025 IC50 = 6 nM T12499 C3FBH0 46891026 IC50 = 8 nM T12499 CYOU90 46891080 IC50 = 4 nM T12499 CJ16KH 46891081 IC50 = 106 nM T12499 C7DOF4 46891082 IC50 = 14 nM T12499 CM14YO 46891147 IC50 = 5 nM T12499 CRPL41 46891148 IC50 = 128 nM T12499 C6FJ7G 46891184 IC50 = 116 nM T12499 C1B2UZ 46891185 IC50 = 546 nM T12499 CYM5B2 46891226 IC50 > 1000 nM T12499 C2DZE0 46891227 IC50 = 209 nM T12499 C1W0JX 46891228 IC50 = 7 nM T12499 CI3VZ0 46891275 IC50 = 699 nM T12499 C28ELR 46912278 Ki = 100 nM T12499 CD4L7V 46912279 Ki = 63.1 nM T12499 C7S2HO 46913757 Ki = 79.43 nM T12499 CT46HI 46913758 Ki = 100 nM T12499 C9PAT7 46927672 IC50 = 10 nM T12499 C60GAV 46929544 IC50 = 385 nM T12499 CHSF07 49806372 IC50 > 1000 nM T12499 C9L3XR 49838879 IC50 = 7000 nM T12499 CRA74I 49842779 IC50 > 10000 nM T12499 CF91RS 49843531 IC50 > 10000 nM T12499 CQ3KU9 50899556 IC50 = 430 nM T12499 C2Y6QS 50938552 IC50 > 10000 nM T12499 C6XYT1 50941838 IC50 > 100000 nM T12499 C61DVY 50990961 IC50 = 610 nM T12499 CV3UP9 50992247 IC50 = 170 nM T12499 CAZQ43 51003133 IC50 = 61 nM T12499 C9NYP4 51036677 IC50 > 10000 nM T12499 C4WRY3 51037112 IC50 > 10000 nM T12499 CRI28Z 51037948 IC50 > 10000 nM T12499 CXA03W 52920796 IC50 = 470 nM T12499 CEQN27 52936621 Ki = 490 nM T12499 C3LB5V 52941849 IC50 = 970 nM T12499 CC42PX 52942070 IC50 = 568 nM T12499 CW2X5E 52944268 IC50 = 20 nM T12499 C9PX2J 52945752 IC50 = 94 nM T12499 CL4ED3 52945753 IC50 = 440 nM T12499 CIR3Q0 52947964 IC50 > 10000 nM T12499 C6OTY5 53251320 IC50 > 19000 nM T12499 CE8OY2 53317913 IC50 < 1 nM T12499 CZ0BV7 53320342 IC50 > 10000 nM T12499 C2W9OA 53324451 IC50 = 4700 nM T12499 CD4H3S 53354074 Ki > 1000 nM T12499 C8NA4L 53384644 IC50 > 30000 nM T12499 CZ1CI3 53469824 IC50 = 741 nM T12499 CXA92G 53484170 IC50 > 20000 nM T12499 C7UK2N 53484181 IC50 > 20000 nM T12499 CKD9H6 53484182 IC50 > 20000 nM T12499 CH05EO 53484183 IC50 = 14114 nM T12499 CAR45T 53484184 IC50 > 20000 nM T12499 CE1ZK6 54759168 IC50 > 10000 nM T12499 C8AB1J 54759606 Ki = 2000 nM T12499 CM8JX1 56604907 IC50 = 10 nM T12499 CN9QD7 56643097 IC50 > 10000 nM T12499 C8GJ9S 56658692 IC50 = 330 nM T12499 CK3A4Z 56658700 IC50 = 3417 nM T12499 C1JD6Z 56658841 IC50 = 603 nM T12499 C98WRJ 56658842 IC50 = 169 nM T12499 C2Z9YO 56662177 IC50 = 4648 nM T12499 CR50XZ 56662178 IC50 = 3208 nM T12499 C8NGC7 56662179 IC50 = 597 nM T12499 C3H0VQ 56662180 IC50 = 945 nM T12499 CWM35E 56662181 IC50 > 20000 nM T12499 CB0VE5 56662182 IC50 > 20000 nM T12499 CEI39Q 56665634 IC50 = 284 nM T12499 CG5K2Q 56665635 IC50 = 365 nM T12499 CVEM27 56665636 IC50 > 20000 nM T12499 CDT3K4 56665637 IC50 > 20000 nM T12499 C9ZTL3 56669088 IC50 > 20000 nM T12499 CC8F0R 56669218 IC50 = 2000 nM T12499 CXW95K 56669219 IC50 = 2262 nM T12499 C8R9TW 56672548 IC50 = 476 nM T12499 C0ROQ7 56672549 IC50 = 10400 nM T12499 CI6K1R 56672550 IC50 > 20000 nM T12499 CC5NQ4 56672551 IC50 = 420 nM T12499 CY0PA7 56672679 IC50 = 722 nM T12499 CP6AE8 56672680 IC50 = 1200 nM T12499 C0GUO4 56672681 IC50 = 70 nM T12499 CWT5X6 56674974 IC50 = 2000 nM T12499 CJA2N4 56675924 IC50 = 1830 nM T12499 C95JAC 56681742 IC50 = 660 nM T12499 CLKP65 56682548 IC50 = 722 nM T12499 CW2YZ7 56682555 IC50 = 539 nM T12499 C1JWN7 56682556 IC50 = 1501 nM T12499 CS9YF2 56682557 IC50 > 20000 nM T12499 COM56E 56682674 IC50 = 3710 nM T12499 CG2A4M 56682676 IC50 = 10 nM T12499 CBOD63 56835089 IC50 > 30000 nM T12499 CI5ZJ7 56835161 IC50 > 100000 nM T12499 CJBL48 56925034 IC50 = 81 nM T12499 CR16SD 56947170 IC50 = 110 nM T12499 CJ47MX 56963907 IC50 = 120 nM T12499 C9L6FD 56963908 IC50 = 3300 nM T12499 CE50IB 56963909 IC50 > 10000 nM T12499 CPHX64 57325478 IC50 > 50000 nM T12499 CQ9BW4 57325479 IC50 > 50000 nM T12499 CE1A9V 57394653 IC50 = 755 nM T12499 CNV76Z 57394656 IC50 = 2790 nM T12499 CD6Y9Z 57395116 IC50 > 30000 nM T12499 C8W6IG 57395117 IC50 > 30000 nM T12499 CG7S0D 57396882 IC50 > 30000 nM T12499 C0UDY9 57401151 IC50 > 30000 nM T12499 CZSM95 57412684 IC50 > 10000 nM T12499 CVK0G4 58056356 IC50 > 50000 nM T12499 CH7L5N 58172700 IC50 = 1448 nM T12499 CWXC70 58180596 IC50 = 1800 nM T12499 C6BPR2 58985201 IC50 > 30000 nM T12499 CZ3TG1 59375154 IC50 = 108 nM T12499 CP9A8T 59503659 IC50 = 271 nM T12499 C1MA6J 59503711 IC50 > 3000 nM T12499 CX29EU 59503744 IC50 = 579 nM T12499 CXJ63M 59603829 IC50 = 37 nM T12499 CQEU96 59603842 IC50 = 3.9 nM T12499 CLH49Z 59790029 IC50 = 3 nM T12499 COH62U 60097413 IC50 > 5000 nM T12499 C1MR8Q 60097495 IC50 > 10000 nM T12499 C9QRX3 60098131 IC50 = 200 nM T12499 CUBL90 66545750 IC50 = 1380 nM T12499 C1HSE0 67035086 IC50 = 690 nM T12499 CWI6K5 67035106 IC50 > 10000 nM T12499 C38RGB 67035556 IC50 = 8900 nM T12499 CV3HW2 67035568 IC50 = 7400 nM T12499 C37NKO 67129970 IC50 = 7790 nM T12499 CK80LJ 67130050 IC50 = 7510 nM T12499 CV63UL 67240318 IC50 > 10000 nM T12499 CZC9M5 67469084 IC50 = 12600 nM T12499 C8I7GC 68293638 IC50 = 8900 nM T12499 CD56XK 68293660 IC50 = 4900 nM T12499 C7GRV2 68755406 IC50 = 3700 nM T12499 C0HA8V 68783839 IC50 = 7 nM T12499 CAIO65 68796885 IC50 = 69 nM T12499 C5DGR9 69036886 IC50 = 818 nM T12499 C7VJ6A 70647728 IC50 = 150 nM T12499 C82FIP 70686752 IC50 = 52 nM T12499 C0QX3Y 70688829 IC50 = 79 nM T12499 CSOT12 70693058 IC50 = 620 nM T12499 CS6NW3 70693059 IC50 = 960 nM T12499 CWM62Q 70694846 Ki = 79.43 nM T12499 C1IEJ2 70789254 IC50 = 113000 nM T12499 C8T7ZP 70789255 IC50 = 20000 nM T12499 COU73Y 71226944 IC50 = 11 nM T12499 C40JOZ 71235465 IC50 = 28 nM T12499 C91HPI 71300299 IC50 > 5000 nM T12499 C2HBG8 71450398 IC50 = 2.35 ug.mL-1 T12499 CKOE90 71451677 IC50 = 1023 nM T12499 CEBO91 71452977 IC50 = 1300 nM T12499 C8AH1B 71454033 IC50 = 12.76 ug.mL-1 T12499 CI37UR 71454035 IC50 = 0.94 ug.mL-1 T12499 CX3AN8 71454037 IC50 > 50 ug.mL-1 T12499 C9ZVW4 71459442 IC50 = 7.91 ug.mL-1 T12499 CO9PR0 71459445 IC50 > 50 ug.mL-1 T12499 CB9V6C 71461186 IC50 = 7.17 ug.mL-1 T12499 CJ6T0K 71462927 IC50 = 4.52 ug.mL-1 T12499 CMV23P 71462929 IC50 = 11.88 ug.mL-1 T12499 C6HF8S 71521082 IC50 = 44620 nM T12499 C9Z3AI 71521083 IC50 = 11050 nM T12499 C5ZKU7 71546969 IC50 = 493 nM T12499 C7ARI9 71547113 IC50 = 617 nM T12499 CCN01X 71547862 IC50 > 10000 nM T12499 C1NPL0 71552941 IC50 > 30000 nM T12499 CA4PS8 71552942 IC50 > 30000 nM T12499 C3UA9C 71553011 IC50 = 15020 nM T12499 CEZ15Y 71553012 IC50 = 1360 nM T12499 CVIA91 71553085 IC50 = 610 nM T12499 C1TR3O 71553152 IC50 = 3680 nM T12499 C7ZR4F 71555873 IC50 = 5 nM T12499 CRX81Q 71575642 IC50 > 10000 nM T12499 CZ31PU 71583657 IC50 = 3200 nM T12499 C3OS8U 71714087 IC50 = 140 nM T12499 C92AZQ 71714088 IC50 = 6050 nM T12499 CN1Y9I 71714230 IC50 = 390 nM T12499 CM6NE9 71714231 IC50 = 50 nM T12499 CG28AP 71714232 IC50 = 120 nM T12499 C91CRY 71714233 IC50 = 1100 nM T12499 C67HDT 71714234 IC50 = 180 nM T12499 CRS05F 71714235 IC50 = 7 nM T12499 CVC19T 71714373 IC50 = 330 nM T12499 CD5C8J 71714374 IC50 = 1100 nM T12499 C51ISR 71714375 IC50 = 360 nM T12499 C5HJK2 71714376 IC50 = 120 nM T12499 C70SJV 71714377 IC50 = 1000 nM T12499 C7E6YV 71720026 IC50 = 264 nM T12499 CF04BD 71765399 IC50 = 6400 nM T12499 CZM1K4 71765510 IC50 = 412 nM T12499 C4KV0T 71765585 IC50 = 1300 nM T12499 C98LKV 71777716 Ki = 440 nM T12499 C3MI4O 71777717 Ki = 55 nM T12499 CD28XR 71816087 IC50 = 2.3 nM T12499 CS10DX 72544168 Ki = 150 nM T12499 CQH45K 72544389 Ki = 110 nM T12499 CMS5O0 72544619 Ki = 1700 nM T12499 CFTK59 72705466 Ki > 25118.86 nM T12499 C1CU0H 72705467 Ki = 15848.93 nM T12499 CX2AW3 72705468 Ki = 100 nM T12499 CVK4Z3 72705469 Ki = 501.19 nM T12499 C4ND6R 72705470 Ki = 100 nM T12499 CT67YO 72706106 Ki = 199.53 nM T12499 C3L2WD 73292576 Ki = 1800 nM T12499 C52LFH 73292907 Ki = 1400 nM T12499 C4FY5U 73346554 Ki = 79.43 nM T12499 CPGD07 73348027 Ki = 2511.89 nM T12499 C05XEV 73348028 Ki = 3162.28 nM T12499 CUW70Y 73348034 Ki = 251.19 nM T12499 CFEU95 73348035 Ki = 501.19 nM T12499 C6K0UL 73348036 Ki = 316.23 nM T12499 CD7X5Q 73348645 IC50 = 360 nM T12499 CD6KE7 73349574 Ki = 19.95 nM T12499 CV8UR4 73351136 Ki = 50.12 nM T12499 CAS60G 73352600 Ki = 125.89 nM T12499 CX75YR 73352604 Ki = 100 nM T12499 C5YKB4 73352605 Ki = 501.19 nM T12499 C03YUP 73355623 Ki = 251.19 nM T12499 CSUZ81 73356106 IC50 = 120000 nM T12499 C6UA4K 73356522 IC50 > 3000 nM T12499 C1A9PR 73357167 Ki = 316.23 nM T12499 CMEV76 74983355 Ki = 340 nM T12499 C0RP9Y 76309810 Ki = 46 nM T12499 C2A7SL 76320747 Ki = 890 nM T12499 CPG3A5 86302574 IC50 > 30000 nM T12499 C1HW4B 89735655 IC50 = 5000 nM T12499 CFB75T 90479825 IC50 = 136 nM T12499 CN7CG9 90644798 IC50 = 142 nM T12499 CLZ71J 90644800 IC50 = 7 nM T12499 C19HKY 90644801 IC50 = 16 nM T12499 C3MU1B 90644802 IC50 = 4 nM T12499 CI0VF7 90644803 IC50 = 4 nM T12499 COA7S0 90644804 IC50 = 4 nM T12499 CY5Z3V 90644805 IC50 = 7 nM T12499 CGIL57 90644806 IC50 = 0.9 nM T12499 CUDB61 90644807 IC50 = 287 nM T12499 CY0UC4 90645194 IC50 > 10000 nM T12499 CE3OV2 90645543 Ki = 1800 nM T12499 CLBC06 90663203 IC50 > 10000 nM T12499 CI8XJ4 90663933 IC50 = 6.24 nM T12499 CMH6T8 90664306 IC50 = 83 nM T12499 CYHR27 91664373 IC50 = 52 nM T12499 C6J0GR 91809511 IC50 = 5900 nM T12499 CAU45T 91971978 IC50 > 30000 nM T12499 CWF97Y 92045039 IC50 = 1220 nM T12499 CY7BI2 118706214 IC50 > 10000 nM T12499 CTP2E8 118737132 Ki = 210 nM T12499 C5GTM2 118737133 Ki = 240 nM T12499 C7MJ5H 118737134 Ki = 640 nM T12499 C3XF2A 118737135 Ki = 600 nM T12499 CNP5K8 118737136 Ki = 660 nM T12499 C8FDR1 118737137 Ki > 2500 nM T12499 C37DUM 121293882 IC50 > 2000 nM T12499 CXQR89 121294143 IC50 > 2000 nM T12499 C08KEM 122179540 IC50 = 2000 nM T12499 CG0RP7 122179547 IC50 = 3000 nM T12499 C1A0SQ 122179548 IC50 = 5200 nM T12499 CLPI09 122180346 IC50 = 13000 nM T12499 CFKD32 122191637 IC50 = 569 nM T12499 C4X7SD 122192466 IC50 > 10000 nM T12499 C8F0DQ 129909860 IC50 = 36 nM T12499 C71KMN 130429150 IC50 = 337 nM T12499 CSG8J3 130429224 IC50 = 77 nM T12499 C5PT1M 130429242 IC50 = 468 nM T12499 C0UNO3 130429244 IC50 = 18 nM T12499 CGFK71 130429248 IC50 = 44 nM T12499 CEX8D1 130429250 IC50 = 137 nM T12499 C9J6ZK 130429255 IC50 = 106 nM T12499 C6OMB1 132204257 IC50 = 425 nM T12499 CV89JM 132231876 IC50 = 420 nM T12499 C6ROQ3 132546210 IC50 = 12 nM T12499 C54FXD 134957362 IC50 > 10000 nM T12499 C1GY2T 135156251 EC50 > 10000 nM T12499 C73DLE 135399258 IC50 = 610000 nM T12499 C1UZW9 135400585 IC50 > 2000000 nM T12499 C6RDV7 135402873 IC50 > 50000 nM T12499 COH41B 135403151 IC50 > 2514000 nM T12499 CR3XN0 135408977 IC50 > 1000000 nM T12499 C7LI1N 135408978 IC50 = 1000 nM T12499 CMB3F6 135409035 IC50 = 200 nM T12499 CHS5X0 135409466 IC50 = 2 ug.mL-1 T12499 C2DH1R 135412832 IC50 = 20 ug.mL-1 T12499 CUI1B3 135417010 IC50 = 1000 nM T12499 CU60YC 135431661 IC50 = 2550 nM T12499 C4VH8I 135438239 IC50 = 600000 nM T12499 C8GZ2B 135449326 Ki = 1200 nM T12499 C5G9XP 135452204 IC50 > 2000000 nM T12499 CX35PB 135468746 IC50 = 500 nM T12499 C9BK5Y 135469311 IC50 = 750000 nM T12499 CWPK94 135478626 IC50 = 40000 nM T12499 CRTS92 135484881 IC50 = 1900000 nM T12499 CZ9L3S 135499405 IC50 = 105000 nM T12499 CTJ48K 135524085 IC50 = 4300 nM T12499 CUT1W7 135524168 IC50 = 6000 nM T12499 CCHD04 135533486 IC50 = 1005000 nM T12499 C3CRI9 135546620 IC50 = 162000 nM T12499 CJ03PU 135566610 IC50 = 162.1 nM T12499 CQ9A5I 135566611 IC50 = 3178.4 nM T12499 C42TOW 135566612 IC50 = 39.2 nM T12499 CN48IF 135566613 IC50 = 203.2 nM T12499 C67IYS 135566618 IC50 = 63.9 nM T12499 CZFA70 135611366 IC50 = 1360 nM T12499 CP54JV 135752285 IC50 = 352000 nM T12499 CX4ZB3 135863110 IC50 > 30000 nM T12499 CYDM01 135891431 IC50 = 0.72 nM T12499 CGI34T 135971386 IC50 = 2.3 nM T12499 CI5U7F 135971387 IC50 = 0.94 nM T12499 CKPA94 135971389 IC50 = 4.8 nM T12499 C3H9ZQ 135971390 IC50 = 2.3 nM T12499 CFT9R7 135971391 IC50 = 0.3 nM T12499 CSO65Z 135971392 IC50 = 1.2 nM T12499 CDS3V4 135971394 IC50 = 0.51 nM T12499 C4X0AQ 135971395 IC50 = 1.5 nM T12499 C45RKA 135971396 IC50 > 100 nM T12499 C36UAJ 135971397 IC50 = 1.5 nM T12499 CR5B1S 135971404 IC50 = 1 nM T12499 C0XP6W 135971405 IC50 = 3.9 nM T12499 C05MXR 135971406 IC50 = 8.2 nM T12499 CNT07W 135971407 IC50 = 0.77 nM T12499 CYZT63 135971410 IC50 = 0.55 nM T12499 C8RV2Z 135971411 IC50 = 0.41 nM T12499 C5HTQ7 135971412 IC50 = 1 nM T12499 CK5Y8N 135971414 IC50 = 0.75 nM T12499 CAKJ23 135971415 IC50 = 1.2 nM T12499 CQ8ZL5 135971416 IC50 = 5.4 nM T12499 CU2V3A 135971417 IC50 = 2.8 nM T12499 CMW4A0 135971418 IC50 = 10 nM T12499 CT8FK6 135971419 IC50 = 0.56 nM T12499 CG2YB1 135971420 IC50 = 1.1 nM T12499 C2K8XA 135971421 IC50 = 0.44 nM T12499 C4GWD2 135971422 IC50 = 3.9 nM T12499 C34CFS 135971423 IC50 = 0.8 nM T12499 C8BJM6 135971424 IC50 = 1 nM T12499 CQ1V2X 135971425 IC50 = 2 nM T12499 CSGD27 135972425 IC50 = 2400 nM T12499 CHA4N2 136013680 IC50 > 10 nM T12499 CP5SD0 136016241 IC50 = 1101.3 nM T12499 C5XIE8 136026041 IC50 = 18000 nM T12499 CIVJ39 136056094 IC50 = 144000 nM T12499 CVIC49 136069671 IC50 = 4800 nM T12499 C48DLS 136123445 IC50 > 1500 nM T12499 CD48LY 136185992 IC50 = 3.75 ug.mL-1 T12499 CPE2B1 136185998 IC50 > 20 ug.mL-1 T12499 CR9XE0 136185999 IC50 = 5 ug.mL-1 T12499 C1I8LC 136186000 IC50 = 5 ug.mL-1 T12499 C40HWO 136186001 IC50 > 20 ug.mL-1 T12499 CK5VW8 136186003 IC50 > 10 ug.mL-1 T12499 C7V1YL 136186004 IC50 > 10 ug.mL-1 T12499 CGP04W 136186009 IC50 = 20 ug.mL-1 T12499 CS5QE7 136186010 IC50 > 20 ug.mL-1 T12499 C1YUD0 136219394 IC50 > 10 nM T12499 CIU8W3 136254389 IC50 > 10 nM T12499 CXC69T 137321158 IC50 = 43 nM T12499 C90FJW 137365215 IC50 = 22 nM T12499 C7ZYL2 137365217 IC50 = 12130 nM T12499 CRKO38 137365218 IC50 = 106 nM T12499 C6K5WV 137365221 IC50 = 1860 nM T12499 C07TXV 137365226 IC50 = 39 nM T12499 CB7N3X 137365228 IC50 = 11600 nM T12499 CMX1A3 137365229 IC50 = 33.5 nM T12499 C42HOT 137365231 IC50 = 54 nM T12499 C1QZH5 137365233 IC50 = 3170 nM T12499 C1OQ7V 137365243 IC50 = 6.5 nM T12499 C5CZ2A 137365245 IC50 = 6 nM T12499 CZOD53 137633880 IC50 = 74 nM T12499 CI1E8V 137634241 IC50 = 699 nM T12499 C7BJY5 137636807 IC50 = 21 nM T12499 CO89DX 137649100 IC50 = 7 nM T12499 CINE03 137652514 IC50 = 100 nM T12499 C28QUP 137652864 IC50 = 194.7 nM T12499 CN0X5D 138454787 IC50 = 860 nM T12499 CLJH31 139209093 IC50 = 42 nM T12499 CI1D9F 139600335 IC50 = 27 nM T12499 CVI30A 139600340 IC50 = 260 nM T12499 C9ZYG8 141366083 IC50 = 910 nM T12499 C6RT5B 142749651 IC50 > 100000 nM T12499 CON17J 142749653 IC50 = 10300 nM T12499 CZ2K6B 142749654 IC50 = 58400 nM T12499 CX2Q5T 142749655 IC50 = 5480 nM T12499 CITW53 142749657 IC50 = 7970 nM T12499 C0TYX5 142749658 IC50 > 100000 nM T12499 CV9WM8 142749660 IC50 > 100000 nM T12499 CF5X8A 142749661 IC50 = 41400 nM T12499 CD1EC9 142749662 IC50 = 17450 nM T12499 CSC02Q 142749664 IC50 > 100000 nM T12499 CNU4M3 145704714 IC50 = 31600 nM T12499 C82RKW 145756290 IC50 = 62 nM T12499 CLU0G7 145756294 IC50 = 225 nM T12499 C6VB3O 145925651 IC50 >= 5000 nM T12499 C9N2TO 145950233 IC50 = 71150 nM T12499 CPZR56 145950296 IC50 = 110 nM T12499 CXQT26 145950509 IC50 = 312 nM T12499 CZ8JC7 145952422 IC50 = 510 nM T12499 C57XVG 145954817 IC50 = 22150 nM T12499 C7AIW6 145957749 IC50 = 130 nM T12499 CDA08X 145957845 IC50 = 502 nM T12499 C9NBS5 145959808 IC50 > 100000 nM T12499 CDNC31 145967951 IC50 < 1 nM T12499 CLUS34 145971460 IC50 = 3300 nM T12499 CF27EG 155511610 IC50 = 1183 nM T12499 C0ZAN6 155512322 IC50 = 250 nM T12499 C0AN1O 155512752 IC50 = 1497 nM T12499 C8TL1A 155513050 IC50 = 26000 nM T12499 C2MD1Q 155513187 IC50 > 10000 nM T12499 CI23DH 155516489 IC50 = 74 nM T12499 CEDI24 155516854 IC50 = 300 nM T12499 C3NA2I 155519537 IC50 = 31 nM T12499 C70NHV 155523393 IC50 > 31000 nM T12499 CS69CA 155532132 IC50 = 40.9 nM T12499 C3LC9I 155536820 IC50 = 1000 nM T12499 C2CG1A 155537016 IC50 > 10000 nM T12499 CKOC12 155537703 IC50 = 10000 nM T12499 CB6AN2 155537880 IC50 = 3980 nM T12499 C3V4LG 155538413 IC50 = 515 nM T12499 CGDJ81 155539793 IC50 = 3100 nM T12499 CDW9G6 155541623 IC50 = 31000 nM T12499 CM8E5L 155548006 IC50 = 3160 nM T12499 CLJ80U 155548662 IC50 = 110 nM T12499 CGTR28 155552797 IC50 = 230 nM T12499 CCV06Q 155554126 IC50 = 120 nM T12499 CZQM57 155554194 IC50 = 3156 nM T12499 CJL3D2 155555429 IC50 = 7940 nM T12499 C3DQI8 155557074 IC50 = 24000 nM T12499 CTR18O 155557674 IC50 = 10000 nM T12499 CVS68Y 155558083 IC50 > 50000 nM T12499 CWD8X0 155558928 IC50 > 31000 nM T12499 CV7H5S 155559048 IC50 = 1000 nM T12499 CT8VX1 155562023 IC50 = 26 nM T12499 CY42EB 155566265 IC50 > 31000 nM T12499 CR6EL3 155568078 IC50 = 34000 nM T12499 C12HQW 155568509 IC50 = 43000 nM T12499 D00DNY 3213 IC50 = 18500 nM T12499 D00ERW 44444843 Ki > 2701 nM T12499 D00HVA 11624601 Ki > 2700 nM T12499 D00RIX 5280443 IC50 = 4 ug.mL-1 T12499 D01IZN 44312289 IC50 = 50000 nM T12499 D01KKU 5281894 IC50 = 80 ug.mL-1 T12499 D01NTW 5328768 IC50 = 7000 nM T12499 D01UYI 5281607 IC50 = 5 ug.mL-1 T12499 D02BUW 2061 IC50 = 3000 nM T12499 D02NNT 53232451 IC50 = 215 nM T12499 D02SRA 44312288 IC50 > 800000 nM T12499 D03AER 9549185 IC50 = 20 nM T12499 D03DZO 11715767 IC50 > 10000 nM T12499 D03NPX 447077 IC50 < 5 nM T12499 D04PEI 11467730 IC50 = 2400 nM T12499 D05FXD 44478401 IC50 = 1.3 nM T12499 D05PTT 5281792 IC50 = 24000 nM T12499 D06HVH 54613583 IC50 > 10000 nM T12499 D06WGX 9549184 IC50 = 147 nM T12499 D07ADX 54764565 IC50 = 333 nM T12499 D07AIB 712152 IC50 < 8 nM T12499 D07ERV 44312580 IC50 = 11000 nM T12499 D07IHM 9823787 IC50 > 10000 nM T12499 D07OXC 11650194 IC50 = 8 nM T12499 D08HFG 24809764 IC50 > 10000 nM T12499 D08LYB 5166 IC50 = 18 nM T12499 D08RZB 11153014 IC50 = 1 nM T12499 D08WOG 9948853 IC50 = 1000 nM T12499 D09DVB 44312287 IC50 = 260000 nM T12499 D09HVH 135566652 IC50 > 10 nM T12499 D09HXU 16086113 IC50 = 94 nM T12499 D09QBA 23378546 IC50 = 6400 nM T12499 D09RYV 9911652 IC50 > 100000000 nM T12499 D09ZNV 447682 IC50 = 11000 nM T12499 D0A2LX 44312363 IC50 = 11000 nM T12499 D0B4PI 44312309 IC50 = 470000 nM T12499 D0B8DE 135469328 IC50 > 10000 nM T12499 D0BS6R 9549183 IC50 = 37 nM T12499 D0D5EW 5311104 IC50 < 5 nM T12499 D0D5KZ 11540659 IC50 = 5 nM T12499 D0D9TU 3894 IC50 = 8000 nM T12499 D0E7VO 59627005 IC50 < 100 nM T12499 D0FH3M 18770833 IC50 > 100000 nM T12499 D0GW4Q 5330524 IC50 < 5 nM T12499 D0H1OK 11562302 Ki = 29.4 nM T12499 D0IR6U 5494425 IC50 > 8000 nM T12499 D0IZ8M 56675928 IC50 = 180 nM T12499 D0M4SY 135440466 IC50 = 341 nM T12499 D0ME9B 46868971 IC50 = 510 nM T12499 D0MF5Y 5281614 IC50 = 4 ug.mL-1 T12499 D0N4LR 53469448 IC50 = 1250 nM T12499 D0O0VZ 667639 IC50 = 20 ug.mL-1 T12499 D0O6OH 71553154 IC50 = 220 nM T12499 D0OH3J 5330526 IC50 < 5 nM T12499 D0OZ2S 11785878 IC50 = 1600 nM T12499 D0P0WT 3139 IC50 > 10000 nM T12499 D0P3JW 447700 IC50 < 5 nM T12499 D0Q2UZ 44312307 IC50 = 260000 nM T12499 D0Q3EW 9549303 IC50 = 131 nM T12499 D0Q3NG 11715520 Ki > 2700 nM T12499 D0QN6U 9806182 IC50 > 10000 nM T12499 D0R2WK 16038120 EC50 > 1000 nM T12499 D0S1KJ 5328733 IC50 < 5 nM T12499 D0S7IE 11658882 Ki > 2700 nM T12499 D0SY6C 5282073 IC50 = 200 ug.mL-1 T12499 D0T8NU 16757525 IC50 > 4000 nM T12499 D0T9FQ 10061448 IC50 > 10000 nM T12499 D0V2LK 10244983 IC50 > 2000000 nM T12499 D0W7LW 44312308 IC50 = 220000 nM T12499 D0Y0BK 11524144 IC50 = 16 nM T12499 D0Y1SR 11844351 IC50 = 2 nM T12499 D0Y4BL 11676971 IC50 = 88 nM T12499 D0Y7HG 5281616 IC50 = 80 ug.mL-1 T12499 D0YZ7H 9797370 IC50 = 100 nM T12499 D0Z4HV 10354294 IC50 > 10000 nM T12499 D0Z7GH 5330525 IC50 < 5 nM T12499 D0Z7TM 22273644 IC50 > 2000 nM T25362 D00SUC 74766595 IC50 = 2300 nM T25362 CI03VK 934 IC50 = 25000 nM T25362 CEQ4V8 2723716 IC50 > 100000 nM T25362 CCYF63 9942424 IC50 = 1258.93 nM T25362 CF47JU 25138011 IC50 = 1100 nM T25362 C68RKH 76310231 IC50 = 31000 nM T25362 CO1EN3 76317452 IC50 = 140 nM T25362 CT5FZ8 76321184 IC50 = 12000 nM T25362 C6XRT0 76321186 IC50 = 37000 nM T25362 CKB5O9 76328366 IC50 = 9100 nM T25362 CUNK03 76335652 IC50 = 9700 nM T25362 CX23ZP 78426670 IC50 > 2500 nM T25362 CKXW73 78427224 IC50 > 2500 nM T25362 CIG3E9 83672127 IC50 = 43000 nM T25362 C2NA5I 91801131 IC50 = 19952.62 nM T25362 CP3DK0 96607511 IC50 = 57 nM T25362 C10RDJ 101882871 IC50 > 100000 nM T25362 C6YT2Q 118598059 IC50 > 4000 nM T25362 C5IZD1 122181577 IC50 > 100000 nM T25362 CRM93S 122181583 IC50 > 100000 nM T25362 CU57QX 122181584 IC50 > 100000 nM T25362 C9QVZ5 122181587 IC50 > 100000 nM T25362 CJQ91K 122181588 IC50 > 100000 nM T25362 C75JVN 122191451 IC50 = 25118.86 nM T25362 C3YX7W 122191453 IC50 = 7943.28 nM T25362 C3IBR8 122191455 IC50 = 7943.28 nM T25362 C59KNQ 122191457 IC50 = 12589.25 nM T25362 CM5X8J 122191459 IC50 = 3162.28 nM T25362 C7ASR0 122191460 IC50 = 10000 nM T25362 CRI6J4 122191461 IC50 = 19952.62 nM T25362 CAS4H6 122191462 IC50 = 50118.72 nM T25362 C9J6LX 122191463 IC50 > 100000 nM T25362 C75NJO 122191464 IC50 > 100000 nM T25362 C50VYK 122191465 IC50 = 31622.78 nM T25362 CSKY20 122191466 IC50 > 100000 nM T25362 CS3L8H 122191467 IC50 = 50118.72 nM T25362 CZ2NV1 122191468 IC50 > 100000 nM T25362 CYTW93 122191469 IC50 > 100000 nM T25362 CZV45H 122191470 IC50 = 31622.78 nM T25362 CF6I2N 122191471 IC50 = 100000 nM T25362 CZU02B 122191472 IC50 > 100000 nM T25362 CE27AS 122191473 IC50 > 100000 nM T25362 CAJ28B 122191475 IC50 = 63095.73 nM T25362 C36PDK 122191476 IC50 = 100000 nM T25362 CQ04FW 122191477 IC50 = 39810.72 nM T25362 C12OHA 122191478 IC50 = 63095.73 nM T25362 CL2K0J 122191479 IC50 = 31622.78 nM T25362 CT6HG3 122191480 IC50 = 50118.72 nM T25362 CK7LD6 122191481 IC50 = 25118.86 nM T25362 CMJ72N 122191482 IC50 = 50118.72 nM T25362 C6H2YQ 122383780 IC50 = 191000 nM T25362 CT2UZ4 125377518 IC50 > 100000 nM T25362 CT4O5U 135567037 IC50 = 11000 nM T25362 CC4H1N 135567038 IC50 = 5700 nM T25362 CQBH95 135567040 IC50 = 33000 nM T25362 CP6IH9 135567041 IC50 = 2300 nM T25362 C8HMG2 135567042 IC50 = 9000 nM T25362 CIW61V 135567106 IC50 = 26200 nM T25362 CL9ZD4 135567108 IC50 = 13900 nM T25362 C1VAI3 135567112 IC50 = 4800 nM T25362 C8LFY7 135567115 IC50 = 6100 nM T25362 C34LUV 137175094 IC50 = 5300 nM T25362 C93YUK 137175210 IC50 = 8300 nM T25362 CYG29R 138393334 IC50 = 2020 nM T25362 CNG82D 138393336 IC50 = 5780 nM T25362 CARJ34 138753212 IC50 = 6130 nM T25362 C4M1EO 155519111 IC50 = 6420 nM T25362 CP8K5E 155540290 IC50 = 5680 nM T25362 CFR06L 155551969 IC50 = 50000 nM T25362 C3SQ4A 155569285 IC50 = 1850 nM T25362 D07IOY 10365 IC50 = 3300 nM T25362 D08IZY 3080614 IC50 = 1995.26 nM T25362 D0S3DD 56963315 IC50 = 39810.72 nM T25362 D0X5US 459617 IC50 = 158.49 nM T16902 D0U2BH 65064 IC50 = 60000 nM T16902 D05HSW 3218 IC50 = 7200 nM T16902 C9XI4U 5703 IC50 = 6100 nM T16902 CL80QG 11820 IC50 = 70000 nM T16902 CHU6D4 343829 IC50 = 221000 nM T16902 C6BCK4 393160 IC50 = 2990 nM T16902 CH6RY3 393161 IC50 = 4430 nM T16902 CSP97B 393162 IC50 = 860 nM T16902 C3Q9OD 393163 IC50 = 4100 nM T16902 C1KX0Y 393164 IC50 = 11800 nM T16902 CT5J0P 393165 IC50 = 12900 nM T16902 CXCB27 393166 IC50 = 5300 nM T16902 COJA52 393167 IC50 = 5710 nM T16902 C2JB3F 393168 IC50 = 1830 nM T16902 CWD08M 393169 IC50 = 15900 nM T16902 CM1L3Q 394797 IC50 = 2720 nM T16902 CCHK53 394798 IC50 = 6510 nM T16902 CHR5Q8 395862 IC50 = 6640 nM T16902 CK69TC 462934 IC50 = 67000 nM T16902 CTIN45 463831 IC50 = 13600 nM T16902 CN7WA6 615185 IC50 = 5400 nM T16902 CEW57U 703058 IC50 = 7660 nM T16902 CO8HA9 832572 IC50 = 12000 nM T16902 C6CQG0 1519964 IC50 = 3690 nM T16902 CJWR09 1561807 IC50 = 67200 nM T16902 CS05BM 1600566 IC50 = 97700 nM T16902 C8E9HY 2221149 IC50 = 34700 nM T16902 C4T8OV 2325816 IC50 = 6190 nM T16902 C1YZ8I 2327942 IC50 = 5770 nM T16902 CS62ZV 2327945 IC50 = 5820 nM T16902 CTVG84 2328663 IC50 = 6010 nM T16902 CNM3K2 2328664 IC50 = 4550 nM T16902 COTE61 2408437 IC50 = 13600 nM T16902 C1LNM0 2467794 IC50 = 6950 nM T16902 CZE13I 2816786 IC50 = 9300 nM T16902 CRIH61 2829592 IC50 = 145900 nM T16902 C5F2BD 2854538 IC50 > 100000 nM T16902 C28JDY 3581192 IC50 = 5000 nM T16902 C2M0BI 5271649 IC50 = 22960 nM T16902 CJ32NW 5276854 IC50 = 1600 nM T16902 C2D4HQ 5337613 IC50 = 5100 nM T16902 C13OPQ 5352088 IC50 = 5000 nM T16902 CK4GM7 7574135 IC50 = 3800 nM T16902 C2FM4R 9875131 IC50 = 1000000 nM T16902 CH41UK 9992116 IC50 = 720 nM T16902 CP96LW 10148995 IC50 > 10000 nM T16902 CY67TD 10197845 IC50 = 3000 nM T16902 CDA2X7 10355152 IC50 = 5030 nM T16902 CUD8X4 10355367 IC50 = 3530 nM T16902 CQMG50 10631053 IC50 = 19952.62 nM T16902 C2QTW8 11052198 IC50 = 28000 nM T16902 CA6X8S 11184436 IC50 = 2200 nM T16902 C61TAS 11230373 IC50 = 203600 nM T16902 C2QXV8 11252989 IC50 = 5400 nM T16902 CR39BD 11253617 IC50 = 5900 nM T16902 C2LGY7 11277137 IC50 = 215100 nM T16902 CC9N1I 11288052 IC50 = 10800 nM T16902 CR0ZW2 11345613 IC50 = 180000 nM T16902 C2NM3S 11357323 IC50 = 34900 nM T16902 C9SOZ5 11379279 IC50 = 125600 nM T16902 C61VWH 11380016 IC50 = 102700 nM T16902 CTL4F6 11390927 IC50 = 77800 nM T16902 CCW1Q4 11402704 IC50 = 7200 nM T16902 C9SLU8 11436521 IC50 = 1600 nM T16902 C0WTI5 12889060 IC50 = 2400 nM T16902 C8XM5J 13017443 IC50 > 10000 nM T16902 CK2NM8 13017478 IC50 > 10000 nM T16902 C7U9KW 13099766 IC50 = 17450 nM T16902 CKF7Z1 13169715 IC50 = 12589.25 nM T16902 C29QHR 13374635 IC50 = 7100 nM T16902 C5S2UI 13554995 IC50 = 4630 nM T16902 C1JO9C 15294640 IC50 > 200000 nM T16902 C1DM9I 18783165 IC50 > 500000 nM T16902 C1XN4F 19425176 IC50 > 10000 nM T16902 CQ14MA 19425177 IC50 = 2500 nM T16902 C4K8PQ 19876167 IC50 = 19800 nM T16902 CBS63Q 21879398 IC50 > 10000 nM T16902 CEOI61 22514828 IC50 = 15100 nM T16902 CPQ68C 33287028 IC50 = 15848.93 nM T16902 C89IXD 33323919 IC50 = 6309.57 nM T16902 C46RLS 42609873 IC50 = 1500 nM T16902 CBJS60 42609916 IC50 = 1800 nM T16902 C31WGD 42609917 IC50 = 5600 nM T16902 CS0D7W 42609918 IC50 = 4900 nM T16902 CNR26A 42609919 IC50 > 10000 nM T16902 C8KC5T 44564008 IC50 > 200000 nM T16902 C6Q7IJ 44564009 IC50 = 19000 nM T16902 C4MOV8 44564010 IC50 = 58000 nM T16902 C8ZBL0 44564011 IC50 > 200000 nM T16902 CC9AP5 44564012 IC50 = 32000 nM T16902 CSN6W0 44564013 IC50 = 102000 nM T16902 CG39PD 44564014 IC50 = 42700 nM T16902 C3KD1U 44564054 IC50 > 200000 nM T16902 CZ1WM3 44564055 IC50 = 3100 nM T16902 CH02PI 44564426 IC50 = 2900 nM T16902 CDV70K 44564427 IC50 = 2900 nM T16902 CN60YA 44564428 IC50 = 2800 nM T16902 CU6I4V 44564429 IC50 = 3200 nM T16902 C2NZU6 44564430 IC50 = 2000 nM T16902 CIA7Q6 44564431 IC50 = 2500 nM T16902 CNKG68 44564432 IC50 = 2600 nM T16902 C3Z9BQ 44564469 IC50 > 10000 nM T16902 CO3UF4 44564514 IC50 = 7500 nM T16902 CL40BF 44564515 IC50 = 109000 nM T16902 CRK2E6 44564516 IC50 = 6500 nM T16902 CT39LN 44564517 IC50 = 162000 nM T16902 C52BJH 44571034 IC50 = 108300 nM T16902 C52ONY 44612934 IC50 > 10000 nM T16902 CFC40W 44612935 IC50 > 10000 nM T16902 C60CBK 44612936 IC50 > 10000 nM T16902 CQZ14C 44612937 IC50 > 10000 nM T16902 CRZ81U 44612938 IC50 > 10000 nM T16902 CSB75V 44612939 IC50 > 10000 nM T16902 CNQL69 44613061 IC50 > 10000 nM T16902 C4VQ2K 44613062 IC50 > 10000 nM T16902 C90VFZ 44613063 IC50 > 10000 nM T16902 C8JL5A 44613064 IC50 > 10000 nM T16902 CX39TE 45256553 IC50 = 11800 nM T16902 CJB6E8 45482638 IC50 = 2600 nM T16902 CYL3P6 45494068 IC50 = 9410 nM T16902 C8K7NG 45882522 IC50 = 6309.57 nM T16902 CC7SL5 46927927 IC50 = 662000 nM T16902 CA80ZD 49653721 IC50 = 41800 nM T16902 C4C0GT 49654128 IC50 = 10700 nM T16902 CG3PR6 52912222 IC50 > 7943.28 nM T16902 C4XCJ0 53257845 IC50 = 25500 nM T16902 C3LX0K 53315396 IC50 = 27900 nM T16902 CQK43N 56662996 IC50 = 86300 nM T16902 C3QZ4C 56666477 IC50 = 4570 nM T16902 C94ZFM 56666478 IC50 = 5900 nM T16902 CBOE48 56669892 IC50 = 6940 nM T16902 CFM97A 56676691 IC50 = 4800 nM T16902 CZH49U 56683381 IC50 = 101000 nM T16902 C2WB3X 56683382 IC50 = 22200 nM T16902 CIPN50 71760902 IC50 > 1000 nM T16902 CO2A1X 71812233 IC50 = 900 nM T16902 CBX37Z 72201043 IC50 = 35000 nM T16902 CX7LT6 76320951 IC50 = 1700 nM T16902 CA7P3H 76320952 IC50 = 2800 nM T16902 CS3W6O 90667751 IC50 = 28800 nM T16902 CZBD29 90667752 IC50 = 78200 nM T16902 CF4W8Q 90667754 IC50 = 63700 nM T16902 C2B4NA 90667755 IC50 = 41800 nM T16902 C9WB3G 95828281 IC50 > 20000 nM T16902 CIX5V3 113222223 IC50 = 15848.93 nM T16902 CX9J1Q 113231872 IC50 = 7943.28 nM T16902 CB5O8P 115579930 IC50 = 31622.78 nM T16902 CVA75B 115611029 IC50 = 1258.93 nM T16902 C21EWV 115611032 IC50 = 15848.93 nM T16902 CM6CX7 118928793 IC50 = 19 nM T16902 CKF18M 118928795 IC50 = 19 nM T16902 CDH8M4 121373418 IC50 > 20000 nM T16902 C47QXT 121376807 IC50 > 20000 nM T16902 C38ERO 121472643 IC50 = 6309.57 nM T16902 C1OIJ9 121476448 IC50 = 501.19 nM T16902 C07JLO 121476460 IC50 = 13 nM T16902 CD3AJ2 126797002 IC50 = 4200 nM T16902 CG9S7A 126961735 Ki = 1.259 nM T16902 CV4D8T 127030247 IC50 = 5000 nM T16902 C0VEM9 131698638 IC50 = 36 nM T16902 CA0P5D 131953422 IC50 = 300 nM T16902 CK1O5N 132153759 IC50 = 70 nM T16902 CGDN94 132275066 IC50 > 20000 nM T16902 CHL8K4 132941768 IC50 = 10000 nM T16902 CU2F1G 135566900 Ki < 3340 nM T16902 CW94QO 136226511 Ki < 3340 nM T16902 C5I9TL 137634095 IC50 = 10000 nM T16902 C2IHE8 137635251 IC50 = 25118.86 nM T16902 CQT3A9 137636309 IC50 > 100000 nM T16902 CULX38 137646779 IC50 = 79.43 nM T16902 CN7V5T 137648161 IC50 = 39810.72 nM T16902 CV7G1I 137654127 IC50 = 6309.57 nM T16902 CSI4V8 137661043 IC50 = 1000 nM T16902 C6C7ZM 138105961 IC50 = 7 nM T16902 C8ZQ2U 141736359 IC50 > 20000 nM T16902 C5VNM4 141736367 IC50 > 20000 nM T16902 C3YGJ5 145948689 IC50 = 300 nM T16902 C96NCH 145950955 IC50 > 20000 nM T16902 C3ZV1O 145952497 IC50 > 20000 nM T16902 CTE74G 145954441 IC50 > 20000 nM T16902 C5WX1Y 145954899 IC50 = 200000 nM T16902 C3D8LO 145955588 IC50 = 160000 nM T16902 CN5YO3 145957310 IC50 > 20000 nM T16902 C8JI5E 145957556 IC50 > 500000 nM T16902 C7C5WL 145958595 IC50 > 20000 nM T16902 C8Z9OM 146205579 IC50 > 20000 nM T16902 CL2SN9 154641364 IC50 = 41 nM T16902 CAN03S 155510571 IC50 = 10 nM T16902 C1E8WH 155513683 IC50 = 17 nM T16902 CAF7V6 155520495 IC50 = 14 nM T16902 C70MDA 155522763 IC50 = 25 nM T16902 C5C6SH 155523656 IC50 = 32 nM T16902 CP4UN7 155523768 IC50 = 35 nM T16902 C98TUC 155526102 IC50 = 47 nM T16902 C5BL1C 155535313 IC50 = 125 nM T16902 C95OQP 155536635 IC50 > 50000 nM T16902 C73HGS 155544332 IC50 = 30 nM T16902 CMON16 155545209 IC50 = 73 nM T16902 C07OQG 155553182 IC50 = 22 nM T16902 C4Z5KF 155562459 IC50 = 30 nM T16902 D03XXT 72201027 IC50 > 20000 nM T16902 D07MTM 403 IC50 > 500000 nM T16902 D07UCF 615184 IC50 = 4200 nM T16902 D08XXD 17815 IC50 = 3600 nM T16902 D09HBR 135566899 Ki = 5520 nM T16902 D0E6JS 167551 IC50 = 5000 nM T16902 D0P0IE 10205 IC50 = 50000 nM T16902 D0W3NA 87642 IC50 = 41910 nM T95736 D0E3TC 44259 IC50 = 2300 nM T95736 D0Z5DM 5081913 IC50 > 100000 nM T95736 CC1PI7 90469 IC50 > 100000 nM T95736 CZ34CV 349435 IC50 = 51000 nM T95736 CFBU18 400433 IC50 = 41000 nM T95736 CYN49L 575802 IC50 = 61100 nM T95736 CU73ST 599501 IC50 > 100000 nM T95736 CL3X6Q 1508801 IC50 > 100000 nM T95736 CMC16L 2782960 IC50 > 100000 nM T95736 CS6VL5 6539018 IC50 > 80000 nM T95736 CK4W6A 8891610 IC50 > 50000 nM T95736 CGRY94 10777396 IC50 > 100000 nM T95736 CACS26 11561968 Ki > 10000 nM T95736 CU0E8O 11690457 Ki > 10000 nM T95736 CB0AP2 11705863 Ki > 10000 nM T95736 CG7X9F 12330558 IC50 > 100000 nM T95736 C78ADF 16751210 IC50 = 1800 nM T95736 C6OY4H 16751569 IC50 = 150 nM T95736 CF0H3L 17229016 IC50 > 100000 nM T95736 CJM4C7 24219848 IC50 > 100000 nM T95736 CC9V2Y 24882562 IC50 = 480 nM T95736 C56VHY 25219675 IC50 > 100000 nM T95736 C90BUF 43157763 IC50 > 100000 nM T95736 CJ7D5T 43157843 IC50 > 100000 nM T95736 C6Z2SA 43560957 IC50 > 100000 nM T95736 CT8P3E 46911431 IC50 = 90000 nM T95736 CVYL83 54768752 IC50 = 24000 nM T95736 CLAQ16 57525824 IC50 = 4.2 nM T95736 C12VDY 58221397 IC50 = 100 nM T95736 C96JRL 58221549 IC50 = 41 nM T95736 CV7E3R 58221661 IC50 = 190 nM T95736 CJS4Y6 58221760 IC50 = 550 nM T95736 C1MR8Q 60097495 IC50 > 10000 nM T95736 CL36SQ 61992242 IC50 > 100000 nM T95736 CNP85L 61992815 IC50 > 100000 nM T95736 CU28AB 62900145 IC50 > 100000 nM T95736 C5L0SQ 68388404 IC50 = 76 nM T95736 CXV8G4 71560537 IC50 = 16000 nM T95736 C57CZF 71560538 IC50 = 4000 nM T95736 CVNT74 71560539 IC50 = 310 nM T95736 CEHS93 71560540 IC50 = 300 nM T95736 C53UOG 71560541 IC50 = 89 nM T95736 CPN3M1 71560660 IC50 = 42000 nM T95736 CLY84V 71560661 IC50 > 80000 nM T95736 CGVE29 71560662 IC50 > 80000 nM T95736 CG9KZ7 71560663 IC50 = 110 nM T95736 C0E9CU 71560664 IC50 = 30000 nM T95736 CB56LM 71560665 IC50 = 70 nM T95736 CW57HX 71560666 IC50 = 2600 nM T95736 C3A1WL 71560667 IC50 = 1200 nM T95736 CG3H8S 71560783 IC50 = 21000 nM T95736 CVBN17 71560784 IC50 = 30000 nM T95736 C7PTA0 71560785 IC50 = 30000 nM T95736 CQ25SH 71580632 IC50 = 63 nM T95736 C1GQE5 71714612 Ki = 41 nM T95736 CPW42O 71714613 Ki = 35.5 nM T95736 C2ZBV7 71714614 Ki = 201 nM T95736 C4GF6B 71714694 Ki = 310 nM T95736 CV50MB 71714695 Ki = 28 nM T95736 CP2LG8 71714710 Ki = 36 nM T95736 CF2U3Z 71714711 Ki = 0.3 nM T95736 C54OCN 71714717 Ki = 101 nM T95736 C3S8AL 71714722 Ki = 20.2 nM T95736 CN31CF 71714729 Ki = 7.5 nM T95736 CUQ0T6 71714731 Ki = 40 nM T95736 CQ8KM1 71715050 Ki = 7 nM T95736 CJ9YX0 71715393 Ki = 3.2 nM T95736 C63JAT 71715396 Ki = 1.5 nM T95736 CK0MZ9 71717636 IC50 = 15000 nM T95736 CE8V7C 71720042 IC50 = 24000 nM T95736 C1XJ2W 71720688 IC50 = 63 nM T95736 CB04OD 82482456 IC50 > 100000 nM T95736 C0ZXY3 86693116 Ki > 250 nM T95736 C0ZOK6 86693155 Ki = 14 nM T95736 CBJ1P2 86693157 Ki = 10 nM T95736 CMY4D7 86693162 Ki = 3.1 nM T95736 CT23XM 86693188 Ki = 0.47 nM T95736 C1H0AG 86693196 Ki = 986 nM T95736 CK8UX7 86693200 Ki = 3 nM T95736 CSKY40 86693215 Ki = 8.7 nM T95736 CAX6M8 86693217 Ki = 4282 nM T95736 CPFS76 86693462 Ki = 9.9 nM T95736 CU78DC 86693540 Ki = 1.7 nM T95736 CWLV65 89754409 Ki = 2503 nM T95736 CU7P5O 89754494 Ki = 2.9 nM T95736 CAO58E 89754729 Ki = 1164 nM T95736 CT04ER 89754780 Ki = 0.9 nM T95736 C2ONT4 89754889 Ki = 405 nM T95736 C2FUO8 89754902 Ki = 0.8 nM T95736 CL4QV3 89754913 Ki = 547 nM T95736 CEI14Q 89754914 Ki = 2 nM T95736 CDEW02 89755037 Ki > 1250 nM T95736 CX0G7V 89755117 Ki = 20 nM T95736 C6Z7ID 89759863 Ki = 0.4 nM T95736 CH75AV 89759865 Ki = 0.8 nM T95736 C1H6FV 117901716 Ki = 68 nM T95736 C0BQS1 117901834 Ki = 1.3 nM T95736 CK8LF5 117902000 Ki = 0.23 nM T95736 CEZW47 117902083 Ki = 0.42 nM T95736 C2GNU7 117902249 Ki = 2 nM T95736 CO5TN3 117902279 Ki = 0.59 nM T95736 C1HX2O 117902381 Ki = 0.07 nM T95736 CYO59C 117902575 Ki = 0.07 nM T95736 CP01MU 117911529 Ki = 4.7 nM T95736 CIOG01 117911755 Ki = 0.86 nM T95736 C1TCH6 117911819 Ki = 16 nM T95736 C98YHE 117911843 Ki = 9.4 nM T95736 C58YIP 117912362 Ki = 0.23 nM T95736 C6TND8 117912488 Ki = 0.18 nM T95736 CPAF91 117923520 Ki = 28 nM T95736 CSY13U 117923525 Ki = 0.08 nM T95736 C5E9JC 117923543 Ki = 0.17 nM T95736 C7WB2P 117923580 Ki = 0.27 nM T95736 CXJ98Z 117923582 Ki = 0.13 nM T95736 CL10MC 117923585 Ki = 0.23 nM T95736 C8LZ6Y 117923640 Ki = 0.05 nM T95736 CB57TM 123132912 Ki = 1280 nM T95736 C3UH2V 129202507 IC50 = 45 nM T95736 C0RE4Q 130270547 IC50 = 1.8 nM T95736 C9G1PS 130270628 IC50 = 21.4 nM T95736 C50DYF 130270664 IC50 = 5.5 nM T95736 C2BE5F 130270736 IC50 = 1.8 nM T95736 CJ1F4A 130270771 IC50 = 4.1 nM T95736 CRV6D7 130270775 IC50 = 2.3 nM T95736 CW5KC8 130270952 IC50 = 1.3 nM T95736 CMX40O 130270954 IC50 = 6.6 nM T95736 CUN4V6 130271143 IC50 = 7.4 nM T95736 C1R6WD 130271145 IC50 = 1.2 nM T95736 CS7ME6 130271227 IC50 = 1.3 nM T95736 C6MZL2 134145793 Ki >= 1250 nM T95736 CQDC40 134151887 Ki = 582 nM T95736 CCH37I 134163557 Ki > 1250 nM T95736 C2AN7T 134611886 IC50 = 8400 nM T95736 CSV6O4 134817242 Ki = 0.3 nM T95736 CKOD92 141758865 IC50 = 189.8 nM T95736 CQJ70P 141758871 IC50 = 85.5 nM T95736 CL04BH 141758877 IC50 = 120 nM T95736 C9S2EO 141758879 IC50 = 2290 nM T95736 CK6E5G 141758883 IC50 = 319 nM T95736 CR0UO6 141758884 IC50 > 10000 nM T95736 CGH4R2 141758885 IC50 = 10910 nM T95736 C01BVU 141758886 IC50 > 10000 nM T95736 CS4W5N 141758888 IC50 = 87.3 nM T95736 CI4AL6 141758890 IC50 = 410 nM T95736 C5REB0 141758892 IC50 = 215 nM T95736 CC1V0S 141758895 IC50 = 11700 nM T95736 CU78RH 141758898 IC50 = 290 nM T95736 CV95IH 141758900 IC50 = 85.2 nM T95736 C4LB2Z 141758901 IC50 = 234 nM T95736 CFH3E1 141758902 IC50 = 2484 nM T95736 C4W8YB 141758903 IC50 = 120 nM T95736 CFW67Y 141758907 IC50 = 641 nM T95736 CCJ30F 141758909 IC50 > 10000 nM T95736 C4Z2HP 141758910 IC50 = 25830 nM T95736 C0EIJ7 141758911 IC50 > 10000 nM T95736 C4J3VR 141758912 IC50 = 3837 nM T95736 C79ZXF 141758918 IC50 > 10000 nM T95736 C69HLJ 141758920 IC50 = 475 nM T95736 CEYA72 141758926 IC50 = 25.7 nM T95736 CVFR90 141758928 IC50 = 2030 nM T95736 C3RO7M 141758929 IC50 = 303 nM T95736 CCIU75 141758930 IC50 = 2204 nM T95736 C0JW8Z 141758931 IC50 = 335 nM T95736 CZH9V1 141758932 IC50 = 219 nM T95736 C1RFW5 141758933 IC50 = 1750 nM T95736 C0OSR6 141758938 IC50 = 204 nM T95736 C4V8EF 141758940 IC50 = 26.1 nM T95736 CH3QM6 141758943 IC50 = 1570 nM T95736 C6JYI1 141758946 IC50 = 468 nM T95736 CC3P2D 141758947 IC50 = 748 nM T95736 C7FYT5 141758948 IC50 = 2060 nM T95736 CE93LI 141758949 IC50 = 22.4 nM T95736 CMWV78 141758951 IC50 = 218 nM T95736 CUV3E7 141758953 IC50 = 2481 nM T95736 C80DZI 141758956 IC50 > 10000 nM T95736 CVBT03 141758957 IC50 > 10000 nM T95736 CZB6J5 141758959 IC50 = 216 nM T95736 CV8YQ9 141758960 IC50 = 290 nM T95736 CEG6I9 141758961 IC50 > 10000 nM T95736 CQT4K6 141758963 IC50 = 720 nM T95736 CDR2I6 141758964 IC50 = 1860 nM T95736 CKXA01 141758965 IC50 = 6160 nM T95736 C3FJN2 141758966 IC50 = 1640 nM T95736 C71BDY 141758967 IC50 = 388 nM T95736 CWF92L 141758969 IC50 = 2061 nM T95736 CJDN92 141758978 IC50 = 6380 nM T95736 CT89FP 145952913 IC50 > 100000 nM T95736 CE6T2K 145965917 Ki = 5.9 nM T95736 C91BHP 145971744 IC50 > 100000 nM T95736 CR73ZD 145976166 Ki = 350 nM T95736 CURX24 145976657 IC50 = 0.8 nM T95736 CML8O0 145979124 IC50 > 100000 nM T95736 CQLH68 145979774 IC50 > 100000 nM T95736 C5YR8W 145979893 IC50 > 100000 nM T95736 CGL48D 145980076 IC50 > 100000 nM T95736 C5LK9A 145980083 IC50 > 100000 nM T95736 CCSY15 145980681 IC50 = 58200 nM T95736 CY80PH 145981483 IC50 = 39600 nM T95736 CN3U5W 145981500 IC50 > 100000 nM T95736 CFSQ94 145981688 IC50 > 100000 nM T95736 CI3P2B 145981824 IC50 > 100000 nM T95736 CVRZ23 145984375 IC50 > 100000 nM T95736 CGE7B8 145987124 IC50 > 100000 nM T95736 C86HGI 145987159 IC50 = 41000 nM T95736 CU3J8R 145987461 IC50 > 100000 nM T95736 CRJQ18 145988918 IC50 > 100000 nM T95736 C8QH2W 145989390 IC50 > 100000 nM T95736 CFAK86 145989643 IC50 > 100000 nM T95736 CHWR01 145989760 IC50 > 100000 nM T95736 C3EIA1 145990026 IC50 > 100000 nM T95736 CBZ94U 145990465 IC50 = 3300 nM T95736 C8M5AU 145990524 IC50 > 100000 nM T95736 C4FQ0C 145990918 IC50 > 100000 nM T95736 CN38UG 145990988 IC50 = 2900 nM T95736 CGSZ75 145991182 IC50 = 24300 nM T95736 C2SY4M 145991367 IC50 > 100000 nM T95736 C0CJ9I 145991401 IC50 > 100000 nM T95736 CI60XK 145991710 IC50 > 100000 nM T95736 C17TOS 145991715 IC50 = 27400 nM T95736 C68ZYI 145991820 IC50 > 100000 nM T95736 C3HIB8 145992014 IC50 = 23000 nM T95736 CF28WP 145992122 IC50 > 100000 nM T95736 C85OWM 145992355 IC50 > 100000 nM T95736 CD54KY 145992596 IC50 > 100000 nM T95736 CQI81V 145992947 IC50 > 100000 nM T95736 C3NU7C 145993088 IC50 > 100000 nM T95736 C0CJ9B 145993626 IC50 = 12500 nM T95736 C2GH5C 145993662 IC50 > 100000 nM T95736 CMJ6G4 145993951 IC50 > 100000 nM T95736 CS61OX 147007484 IC50 = 5.9 nM T95736 CXN9Z8 155510685 IC50 = 2230 nM T95736 C7H5XM 155517858 IC50 = 9.1 nM T95736 CJP09I 155520168 Ki = 0.16 nM T95736 CS29GT 155528718 Ki > 1250 nM T95736 C0FAD1 155540387 Ki > 1250 nM T95736 CLA0I9 155552645 Ki = 634 nM T95736 D07MQC 9949093 IC50 > 100000 nM T95736 D0J3LR 11634725 Ki > 5000 nM T95736 D0LE7J 58221375 IC50 = 20 nM T95736 D0P0IE 10205 IC50 > 100000 nM T65721 C43DAY 68635 IC50 = 4600 nM T65721 C5KW4H 72311 IC50 = 7000 nM T65721 CYUH56 363208 IC50 = 31000 nM T65721 CWJ43S 443767 IC50 = 34000 nM T65721 CORM47 1849091 IC50 = 21300 nM T65721 C9N5XB 2026662 IC50 = 8700 nM T65721 CD8BS4 2999946 IC50 = 46100 nM T65721 CYZ0U7 4891910 IC50 = 5300 nM T65721 CAK90T 4893331 IC50 = 27900 nM T65721 CU8LQ0 4893774 IC50 = 24200 nM T65721 CF9QP2 9076354 IC50 = 24100 nM T65721 CT8RA9 9099810 IC50 = 57200 nM T65721 CK7N4D 9880653 IC50 = 2700 nM T65721 CD57RY 24344410 IC50 = 28300 nM T65721 CN3Y9K 25138381 IC50 = 9300 nM T65721 CDU76N 25164618 IC50 = 54000 nM T65721 C4OP0C 25165019 IC50 = 58000 nM T65721 C51DAH 45272995 IC50 = 12200 nM T65721 CP57CD 45483073 IC50 = 13000 nM T65721 CURM73 51031035 IC50 = 1100 nM T65721 C0EQA8 90655048 IC50 = 95000 nM T65721 C1KBS9 135431654 IC50 = 1800 nM T65721 C9PY6U 135959764 IC50 = 37000 nM T23984 CG3PR6 52912222 IC50 > 1.259 nM T23984 CIPN50 71760902 IC50 > 1000 nM T23984 COZ8S1 78319129 IC50 > 1000 nM T23984 CYX7T2 117072549 IC50 = 3410 nM T23984 C87ZPY 118796358 IC50 = 117 nM T23984 CC14FI 118933132 IC50 = 82 nM T23984 C9MQF0 119098887 IC50 = 240 nM T23984 C0QX4D 119098889 IC50 = 108 nM T23984 CGA71L 127048256 IC50 = 3283 nM T23984 CH6T5J 127048257 IC50 = 2976 nM T23984 C60SZQ 127048258 IC50 = 4307 nM T23984 C50BMV 127049279 IC50 = 230 nM T23984 CTF4N2 127051087 IC50 = 188 nM T23984 CLSZ47 127051725 IC50 = 41 nM T23984 CMY93U 127051726 IC50 = 3725 nM T23984 CY8V1A 127051727 IC50 = 1565 nM T23984 CXZT48 127052023 IC50 = 2475 nM T23984 CV4X7R 135566898 Ki = 3540 nM T23984 CU2F1G 135566900 Ki < 1430 nM T23984 CW94QO 136226511 Ki < 1430 nM T23984 CQT3A9 137636309 IC50 > 100000 nM T23984 CQ6XB7 139030526 IC50 = 63095.73 nM T23984 D08LXU 91827372 IC50 = 3300 nM T23984 D09HBR 135566899 Ki = 2720 nM T23984 D0O6XT 91827373 IC50 = 140 nM T17067 C4DQ7P 11222830 IC50 = 3000 nM T17067 C3Z5CV 46830074 IC50 > 200000 nM T17067 D0N6BC 950368 Ki = 100000 nM T17067 D0Y7OI 11563133 Ki = 4000 nM T07663 D05MQK 110635 IC50 = 1.2 nM T07663 D0C9SY 135400189 Ki = 0.7 nM T07663 D0F9GE 3108 IC50 = 574 nM T07663 D0NJ3V 4680 IC50 = 8800 nM T07663 D0Y5JC 9869929 Ki = 5 nM T07663 D0Y9ZE 4197 IC50 = 740 nM T07663 D0Z7ZM 135398744 Ki = 1.6 nM T07663 D03QJL 3671 IC50 = 103000 nM T07663 D05OQG 5318997 IC50 = 5900 nM T07663 D09OCK 135430955 IC50 = 4.2 nM T07663 D0A9IY 135564558 IC50 > 10000 nM T07663 D0L0BX 5318980 IC50 = 2200 nM T07663 D0M9FQ 11465695 IC50 = 0.5012 nM T07663 D0T5PO 5092 IC50 = 720 nM T07663 D05VBJ 71295299 IC50 > 10000 nM T07663 D0WS3T 72706254 IC50 = 260 nM T07663 D00SPK 23665864 IC50 = 3.7 nM T07663 D00YPW 135399235 Ki = 130 nM T07663 D01QUF 9842576 Ki > 100000 nM T07663 D02EMR 151170 IC50 > 10000 nM T07663 D05VLN 55690 IC50 = 58000 nM T07663 D0BK6B 3021729 IC50 > 10000 nM T07663 D0F0CS 5723 IC50 > 10000 nM T07663 D0K2BQ 71356 Ki = 7500 nM T07663 D0N5SC 135536943 IC50 = 1.23 nM T07663 D0W8OH 135529458 IC50 = 80 nM T07663 CVQ0G5 1348 IC50 = 500 nM T07663 C03NGJ 1713 IC50 = 230 nM T07663 CH8J2B 4977 Ki = 600000 nM T07663 CCJ8F0 5353 IC50 = 21000 nM T07663 C3B8VG 5369 IC50 = 1 nM T07663 CAMB41 100554 IC50 = 5500 nM T07663 C9T3FB 105007 IC50 = 1580 nM T07663 CGA17S 127779 Ki = 6500 nM T07663 C1H8NR 155248 IC50 > 50000 nM T07663 CH2P8A 158961 Ki = 600000 nM T07663 CVN23X 158962 Ki = 600000 nM T07663 CL27HC 160179 IC50 = 9300 nM T07663 CYWS98 185848 IC50 > 40000 nM T07663 C78DLE 205964 IC50 = 360 nM T07663 C1B6ZL 662965 IC50 > 50000 nM T07663 C3A4HW 675226 IC50 = 8600 nM T07663 CA56MW 675227 IC50 = 3900 nM T07663 CHAB75 696516 IC50 = 1900 nM T07663 CW2U6N 698956 IC50 = 420 nM T07663 CYBA13 719250 IC50 = 4700 nM T07663 C1HM0K 832282 IC50 = 4300 nM T07663 C9KVI7 832283 IC50 = 22000 nM T07663 CM6Q1D 869895 IC50 = 2400 nM T07663 C6QBR5 874599 IC50 = 540 nM T07663 CR7A3U 930420 IC50 = 1200 nM T07663 CWIA36 987187 IC50 = 5600 nM T07663 CT62PH 987189 IC50 = 3100 nM T07663 CO0Z8N 1002275 IC50 = 1700 nM T07663 CXQ4P8 1183964 IC50 = 860 nM T07663 CZQ09F 1204882 IC50 = 7200 nM T07663 CHP0S3 1204883 IC50 = 570 nM T07663 C0JM2Q 1215407 IC50 = 700 nM T07663 CZ2XI5 1271431 IC50 = 3100 nM T07663 COW58U 1277329 IC50 = 190 nM T07663 C6VF0S 1490272 IC50 = 840 nM T07663 CQ69OY 1490552 IC50 = 1100 nM T07663 CD0G9E 1553819 IC50 = 14000 nM T07663 CYD6E3 1553838 IC50 = 190 nM T07663 CXP17G 1604254 IC50 = 4600 nM T07663 C8JLO0 2243267 IC50 = 370 nM T07663 CTQ23N 2452792 IC50 = 800 nM T07663 CLNU08 2456309 IC50 = 740 nM T07663 CYP23V 2465033 IC50 = 800 nM T07663 CE70KT 2471983 IC50 = 1200 nM T07663 CE4D1W 2789492 IC50 = 5600 nM T07663 CFC30O 2789499 IC50 = 1000 nM T07663 C4LSR7 2886111 IC50 > 10000 nM T07663 C6AT3L 2930929 IC50 = 6300 nM T07663 CD70ZG 3119958 IC50 = 8700 nM T07663 C4MSC9 3120507 IC50 = 3000 nM T07663 CPX4V3 4352680 IC50 = 130620 nM T07663 C5IZS9 4636426 IC50 = 746450 nM T07663 CC3LA4 4672917 IC50 = 8500 nM T07663 C5P0LU 4672918 IC50 = 29300 nM T07663 C3JHM8 4687521 IC50 = 1.2 nM T07663 C0JVX6 4867627 IC50 = 4900 nM T07663 CN0Z3D 4880961 IC50 = 11000 nM T07663 C0C9HP 6610310 IC50 = 19 nM T07663 CAYS61 6918354 IC50 = 4000 nM T07663 CB40PM 6918356 IC50 = 200 nM T07663 CI7K0P 6918667 IC50 = 69800 nM T07663 CP1GO7 6918668 IC50 > 84900 nM T07663 CA05PF 6918674 IC50 = 700 nM T07663 C87WYR 6918795 IC50 > 67300 nM T07663 CRGE51 6918796 IC50 > 101000 nM T07663 CUP4M8 6918797 IC50 > 50700 nM T07663 C0LRO8 6918798 IC50 > 101000 nM T07663 C53ESK 6918799 IC50 > 91000 nM T07663 CU1E0G 6918800 IC50 > 101000 nM T07663 CRU46D 7161211 IC50 = 3250 nM T07663 CQ41MA 8055545 IC50 = 2300 nM T07663 CZF0N3 8055573 IC50 = 2400 nM T07663 CN86QP 8078832 IC50 = 2500 nM T07663 CI15SH 9797222 IC50 = 14000 nM T07663 CNC2F4 9798336 IC50 > 1000000 nM T07663 CFJ62Y 9799389 IC50 > 10000 nM T07663 CZH08Y 9802738 IC50 = 7.2 nM T07663 CDV76T 9803328 Ki = 0.29 nM T07663 CR09LM 9805655 IC50 = 0.3 nM T07663 CB57DJ 9807085 IC50 = 72 nM T07663 CXF0J7 9818343 IC50 = 10 nM T07663 C1CXA5 9818702 IC50 = 5000 nM T07663 CSOX21 9819114 IC50 = 2.8 nM T07663 C1MN3A 9821924 IC50 = 2 nM T07663 C7FY1U 9824408 IC50 = 1.1 nM T07663 C4J2XE 9836643 IC50 > 101000 nM T07663 C4YB1S 9844037 IC50 = 5.3 nM T07663 C5YQB0 9859898 IC50 = 78000 nM T07663 CZGM43 9864862 IC50 = 22000 nM T07663 CEI5P4 9868140 IC50 = 440 nM T07663 C92GMV 9879320 IC50 = 13000 nM T07663 C0Q5VN 9880010 IC50 > 101000 nM T07663 CWD1F6 9880288 IC50 > 101000 nM T07663 C2NK8E 9888568 IC50 = 0.56 nM T07663 C0P8ZH 9892886 Ki = 0.21 nM T07663 CC05QE 9901606 IC50 = 101000 nM T07663 CMBO89 9912467 IC50 = 2000 nM T07663 CBA29H 9922545 IC50 > 101000 nM T07663 CKF4C2 9922691 IC50 = 73200 nM T07663 CY17NM 9922999 IC50 = 8400 nM T07663 C70AMC 9924305 IC50 = 7270 nM T07663 CKI6N2 9924468 IC50 > 88000 nM T07663 C6AZ5F 9924709 IC50 > 101000 nM T07663 C54ICU 9927654 IC50 = 3500 nM T07663 C60BWM 9933503 IC50 = 0.8 nM T07663 CX1UV7 9946954 IC50 = 20160 nM T07663 C7OP5A 9947052 IC50 = 3970 nM T07663 C04HAV 9949594 IC50 = 225 nM T07663 C53AVJ 9951793 IC50 = 2.3 nM T07663 CE8ZD7 9954790 IC50 = 0.93 nM T07663 CH46TF 9954942 Ki = 0.23 nM T07663 C8X7RN 9956576 IC50 = 0.1 nM T07663 C2OYA1 9957043 IC50 = 0.55 nM T07663 CJO0X4 9966737 IC50 = 10940 nM T07663 CFP1Y5 9966830 IC50 > 101000 nM T07663 C9NKY4 9967652 IC50 = 74000 nM T07663 CI6AX1 9968005 IC50 > 101000 nM T07663 C7PCS8 9968050 IC50 = 40350 nM T07663 CFB48Q 9968370 IC50 = 98000 nM T07663 CU73AJ 9968471 IC50 > 101000 nM T07663 C0AP8O 9969020 IC50 = 17880 nM T07663 C9X7PF 9972372 IC50 = 8800 nM T07663 CL6V2I 9973407 IC50 = 770 nM T07663 CCDX84 9973586 IC50 = 0.53 nM T07663 C5AE2I 9973597 IC50 > 200000 nM T07663 CTQ59Y 9975543 IC50 = 3600 nM T07663 CW3S7O 9977675 IC50 > 1000000 nM T07663 C05RPA 9977814 IC50 = 2700 nM T07663 C20XIY 9985391 IC50 = 2200 nM T07663 CHG4K5 9992525 IC50 = 64000 nM T07663 CO87TV 9994528 IC50 = 100 nM T07663 CC86WM 9995163 IC50 = 6800 nM T07663 CB9EY5 9995187 IC50 = 90 nM T07663 CWJ0K5 9995367 IC50 = 210 nM T07663 CZR07N 9995467 IC50 = 930 nM T07663 C3GHJ7 9996490 IC50 = 105 nM T07663 CH70VI 9996675 IC50 = 1100 nM T07663 CE5O4D 9998316 IC50 = 350 nM T07663 CYS20P 10004422 IC50 = 38000 nM T07663 CB41WF 10017397 IC50 = 3000 nM T07663 CKE92N 10017795 IC50 = 3600 nM T07663 CHJ73C 10018556 IC50 = 8700 nM T07663 CI9WK7 10021158 IC50 = 1300 nM T07663 C6MUC5 10024867 IC50 = 2500 nM T07663 C5E4QJ 10030897 Ki = 0.24 nM T07663 C1G5XC 10032458 IC50 = 6500 nM T07663 CE25WO 10039122 IC50 = 4400 nM T07663 CUYW65 10039809 IC50 = 20000 nM T07663 C0SZB8 10039848 IC50 = 36300 nM T07663 CJ1Q7Z 10040540 IC50 = 50 nM T07663 CJ05CZ 10040882 IC50 = 15000 nM T07663 CK5VB0 10041530 IC50 = 14000 nM T07663 C9FD1X 10041853 IC50 = 7500 nM T07663 CT6Y9J 10043209 IC50 > 1000000 nM T07663 CY6FQ4 10053217 IC50 = 3 nM T07663 CD1N4K 10062262 IC50 = 1000 nM T07663 CHCJ86 10065791 IC50 = 810 nM T07663 CC6PO8 10066654 IC50 > 40000 nM T07663 C3MA2L 10067044 IC50 > 1000000 nM T07663 C5FCT6 10070215 IC50 = 0.6 nM T07663 COSV65 10074226 Ki = 0.23 nM T07663 CG39NX 10083598 IC50 = 40000 nM T07663 C5P7AS 10083609 IC50 = 6000 nM T07663 C7YBR0 10083610 IC50 = 33000 nM T07663 CAX67L 10084334 IC50 = 3000 nM T07663 CP6W8T 10086869 IC50 = 18500 nM T07663 CLB5S6 10087203 IC50 = 11000 nM T07663 CNA75V 10087755 IC50 = 1400 nM T07663 CJ16FV 10087963 IC50 > 1000000 nM T07663 CSP05N 10088555 IC50 = 730 nM T07663 CRW6E1 10088941 IC50 > 40000 nM T07663 C09ZNQ 10088960 IC50 = 2.6 nM T07663 C0O6MQ 10089225 IC50 = 2300 nM T07663 C13QUP 10089597 IC50 = 65000 nM T07663 CARY56 10091146 IC50 > 200000 nM T07663 CP8I5O 10093297 IC50 = 9800 nM T07663 CS4QG0 10095269 IC50 = 900 nM T07663 C61QRH 10096810 IC50 = 49000 nM T07663 CN23KJ 10105662 IC50 = 18000 nM T07663 CP3D7N 10108060 IC50 = 6000 nM T07663 C12LED 10109572 IC50 > 101000 nM T07663 CT0A4J 10113055 IC50 = 9 nM T07663 CPWL59 10113972 IC50 = 8 nM T07663 C5GRV3 10117157 IC50 = 56 nM T07663 C2PBD6 10131447 IC50 = 19300 nM T07663 C3AOI5 10138533 IC50 = 134 nM T07663 C8XPO7 10145438 Ki = 0.2 nM T07663 C4F3SH 10151707 IC50 = 1.585 nM T07663 C3H1IG 10161792 IC50 = 750 nM T07663 C89DXP 10181676 IC50 = 6 nM T07663 C5HC2X 10182563 IC50 = 52400 nM T07663 CK3TY8 10187239 IC50 = 2.089 nM T07663 CJZK81 10195399 IC50 = 1.9 nM T07663 C3GN8K 10200432 IC50 > 101000 nM T07663 CK81LJ 10203901 Ki = 4 nM T07663 CEY6F7 10205437 IC50 = 10.96 nM T07663 CLW92Y 10205894 IC50 = 65 nM T07663 CULN70 10206649 Ki = 0.31 nM T07663 C8JR4W 10221093 IC50 = 44000 nM T07663 CFGO46 10221904 IC50 = 60000 nM T07663 C8V6FE 10225063 IC50 = 2 nM T07663 CX35CL 10244508 IC50 = 6200 nM T07663 CGA50J 10244709 IC50 = 230 nM T07663 CT7RC0 10245770 IC50 = 15000 nM T07663 CC80XO 10247363 IC50 = 620 nM T07663 CP4YR0 10248176 IC50 > 1000000 nM T07663 C8G3BJ 10249105 IC50 = 3.5 nM T07663 C7MQZ1 10249183 IC50 > 1000000 nM T07663 C3AFN6 10250999 IC50 = 8300 nM T07663 CRK1U0 10252045 IC50 = 53000 nM T07663 C7GTC0 10264205 IC50 = 3020 nM T07663 C5VQL9 10264224 IC50 = 26000 nM T07663 CP70US 10267904 IC50 = 13800 nM T07663 CQ61CV 10268304 IC50 = 68400 nM T07663 C1QU2B 10268305 IC50 = 9470 nM T07663 C1VL9A 10269511 IC50 = 0.48 nM T07663 CH9C4K 10269859 IC50 = 23600 nM T07663 CR92JY 10270352 IC50 > 101000 nM T07663 C7CHR0 10270536 IC50 = 12600 nM T07663 C1VH6L 10279632 Ki = 8 nM T07663 C1FA4P 10288830 IC50 = 1.6 nM T07663 C3YO7N 10289243 IC50 = 1.288 nM T07663 CISQ36 10291967 IC50 = 63000 nM T07663 CKR74B 10292282 IC50 = 840 nM T07663 CA54BI 10294138 IC50 = 4 nM T07663 CKQ8I4 10313609 IC50 = 860 nM T07663 CUE72P 10314633 IC50 = 16 nM T07663 CJO72N 10315684 IC50 = 14 nM T07663 CIPN48 10316358 IC50 = 22000 nM T07663 C36AGZ 10321525 IC50 = 240 nM T07663 C90QZM 10324834 IC50 = 2.1 nM T07663 CRJW04 10334696 IC50 = 4000 nM T07663 C5K1LH 10336744 IC50 = 480 nM T07663 C6AQ0U 10338401 IC50 > 200000 nM T07663 C4GB5L 10338602 IC50 = 38 nM T07663 C52EPV 10339653 IC50 > 1000000 nM T07663 CMJG73 10342601 IC50 = 1200 nM T07663 CK05FV 10343476 IC50 = 68000 nM T07663 C32IUF 10344870 IC50 = 40000 nM T07663 CHZL20 10345264 IC50 = 1.6 nM T07663 CA18KO 10347662 IC50 = 20000 nM T07663 CC4W3M 10349233 IC50 = 24000 nM T07663 CQD9O7 10355498 IC50 = 6000 nM T07663 C4BL9Q 10358104 IC50 = 20000 nM T07663 CG8V6F 10358836 IC50 = 9000 nM T07663 CEIW08 10359077 IC50 = 175000 nM T07663 CP5S1A 10359273 IC50 = 165 nM T07663 C7QYK3 10359377 IC50 = 2150 nM T07663 CR35FX 10378878 IC50 = 15000 nM T07663 C2H9SE 10380126 IC50 = 4000 nM T07663 C6E5OY 10380621 IC50 = 5900 nM T07663 C5EVH3 10381520 IC50 = 380 nM T07663 C0J7OV 10382041 IC50 = 11000 nM T07663 C9IK3H 10382413 IC50 = 120 nM T07663 C52DNX 10384462 IC50 = 5500 nM T07663 CF6A1Q 10385088 IC50 > 200000 nM T07663 CZ6X9Y 10391444 IC50 = 3100 nM T07663 CQOX84 10393352 IC50 = 3.5 nM T07663 C9-APR-07 10394586 IC50 = 34000 nM T07663 CI8B3P 10401473 IC50 = 1000 nM T07663 C6E0PG 10401818 IC50 = 2000 nM T07663 C7X4EW 10402019 IC50 = 630 nM T07663 C78SRU 10403787 IC50 = 72 nM T07663 CUF0X6 10404302 IC50 > 1000000 nM T07663 C0ADP3 10404378 IC50 = 56000 nM T07663 CV3I5E 10405045 IC50 = 380 nM T07663 CP8ZV5 10408375 IC50 = 140 nM T07663 C4BF5Y 10411270 IC50 = 1.4 nM T07663 CQUE27 10413015 IC50 = 37000 nM T07663 CS7J4V 10414339 IC50 = 16 nM T07663 C0ZLB5 10423102 IC50 = 1000 nM T07663 C5ZQG3 10426854 IC50 = 5500 nM T07663 C5HMX2 10428149 IC50 = 32000 nM T07663 CB2X9W 10429802 IC50 = 110 nM T07663 CAW23H 10434818 IC50 > 1000000 nM T07663 CH76CS 10443650 IC50 = 42000 nM T07663 CBH5V4 10445800 IC50 = 24000 nM T07663 CZ8IC4 10448177 IC50 > 1000000 nM T07663 CYU38H 10448853 IC50 = 1600 nM T07663 C1RZ9E 10449000 IC50 > 1000000 nM T07663 C18EHX 10449737 IC50 = 1300 nM T07663 CU2HN6 10450290 IC50 > 200000 nM T07663 C9IF7Y 10451065 IC50 = 4.8 nM T07663 CY4O0K 10452443 IC50 = 38000 nM T07663 CI1H7F 10452463 IC50 = 0.05 nM T07663 C4LOK1 10454517 IC50 = 3600 nM T07663 CR04LJ 10456913 IC50 = 54000 nM T07663 CASV91 10466228 IC50 = 34000 nM T07663 C6IP3N 10468291 IC50 = 24000 nM T07663 C6PXC2 10471556 IC50 = 31 nM T07663 C2FYT6 10471617 IC50 = 2300 nM T07663 C2DEO3 10472374 IC50 > 200000 nM T07663 CBMI84 10473521 IC50 = 810 nM T07663 CF0I6O 10479155 IC50 = 13000 nM T07663 C5CI3G 10479468 IC50 = 53000 nM T07663 CZ92DR 10481735 IC50 = 9 nM T07663 CE2RJ7 10499713 IC50 = 420 nM T07663 C0N5LU 10504068 IC50 = 0.53 nM T07663 C71AJB 10520277 IC50 = 19 nM T07663 CSZ7L0 10520799 IC50 = 19 nM T07663 CPWU60 10524067 IC50 = 8000 nM T07663 CG1QK8 10542139 IC50 = 6200 nM T07663 C7LG4O 10543051 IC50 = 26000 nM T07663 C7K5PG 10544204 IC50 = 26 nM T07663 C0Z1CT 10546352 IC50 = 63 nM T07663 CCK5F8 10549901 IC50 = 120 nM T07663 CMK39Q 10553487 IC50 = 200 nM T07663 CQW79N 10554042 IC50 = 10000 nM T07663 CTYQ03 10565296 IC50 = 7500 nM T07663 C1DO9H 10573238 IC50 = 275 nM T07663 CI8GS1 10574005 IC50 = 590 nM T07663 CY9P5W 10575733 IC50 = 30000 nM T07663 CFY5J3 10576937 IC50 = 305 nM T07663 CYD4Z2 10592106 IC50 = 140 nM T07663 C4HVR8 10595830 IC50 = 5600 nM T07663 CRKT15 10597744 IC50 = 43 nM T07663 C71YLE 10598277 IC50 = 4 nM T07663 CJ7CU4 10603606 IC50 = 1000 nM T07663 CR9H4Z 10617782 IC50 = 4500 nM T07663 CK3GR5 10624131 IC50 = 20000 nM T07663 C25WRZ 10627119 IC50 = 9000 nM T07663 CC68NQ 10636956 IC50 = 100 nM T07663 CE57IW 10639502 IC50 = 3300 nM T07663 C0U8KD 10642598 IC50 = 10000 nM T07663 CX61NW 10642809 IC50 = 810 nM T07663 CNK65G 10646809 IC50 = 100000 nM T07663 CKNA14 10648008 IC50 = 20000 nM T07663 C32TRJ 10659857 IC50 = 240 nM T07663 C9GJ5K 10660011 IC50 = 13000 nM T07663 C8KWM5 10663015 IC50 = 34 nM T07663 CP13SC 10663562 IC50 = 80 nM T07663 COQ17R 10666144 IC50 = 9200 nM T07663 CBQ24O 10668762 IC50 = 4000 nM T07663 C1R9VY 10669652 IC50 = 110 nM T07663 CB9Y7A 10669693 IC50 = 40000 nM T07663 CWYZ15 10670833 IC50 = 2 nM T07663 C2Y5HF 10675032 IC50 = 800 nM T07663 CW12SY 10690095 IC50 = 510 nM T07663 CV6WT3 10692240 IC50 > 30000 nM T07663 C29YKI 10692613 IC50 = 1200 nM T07663 C0FPL8 10692684 IC50 = 800 nM T07663 CI6ON5 10698519 IC50 = 4000 nM T07663 C2JTX7 10715358 IC50 = 400 nM T07663 C1I8VM 10716045 IC50 = 1500 nM T07663 CDMP96 10717370 IC50 = 30000 nM T07663 CCI8R7 10729204 IC50 > 100000 nM T07663 C2P5VY 10731865 IC50 = 610 nM T07663 CSQG30 10741916 IC50 = 0.55 nM T07663 CTCS25 10753773 IC50 = 100 nM T07663 C3X8UM 10754735 IC50 = 800 nM T07663 C4EG9Z 10759241 IC50 = 19 nM T07663 CEIZ87 10761565 IC50 = 54 nM T07663 CINX82 10763354 IC50 = 20000 nM T07663 COVG15 10764868 IC50 = 120 nM T07663 C51XRM 10776762 IC50 = 2400 nM T07663 CR4O8B 10781567 IC50 = 16000 nM T07663 C7O8WB 10787783 IC50 = 180 nM T07663 CLM42P 10788651 IC50 = 20000 nM T07663 C7U2NT 10808382 IC50 = 140 nM T07663 CEI0J8 10809340 IC50 = 49 nM T07663 CDF43L 10810826 IC50 = 66 nM T07663 CTMX70 10815441 IC50 = 58000 nM T07663 CA9UW6 10816539 IC50 = 200 nM T07663 C5V1AY 10828080 IC50 = 60 nM T07663 C0SEG5 10830345 IC50 = 6000 nM T07663 CI0XH5 10833134 IC50 = 98 nM T07663 CT6VP3 10834312 IC50 = 560 nM T07663 C8HY0A 10835448 IC50 = 11 nM T07663 CZY5K8 10836947 IC50 = 600 nM T07663 CG2O1B 10836974 IC50 = 200 nM T07663 CR50XV 10841036 IC50 = 40000 nM T07663 CJ0TR9 10854527 IC50 = 100 nM T07663 CW3T1L 10863491 Ki = 154 nM T07663 C9TH7M 10863695 Ki = 1.75 nM T07663 CH0B6V 10885231 Ki = 188 nM T07663 CQ8YB7 10897309 Ki = 1.78 nM T07663 C0RTU9 10897531 EC50 = 9.5 nM T07663 CG0LM2 10907083 Ki = 0.4 nM T07663 CB6U4L 10929261 Ki = 0.47 nM T07663 CL1RW3 10929391 Ki = 0.21 nM T07663 C0BS9L 10939795 Ki = 0.71 nM T07663 C4KLI7 10951390 Ki = 1.14 nM T07663 C9UXZ6 10951441 Ki = 1.01 nM T07663 CP59RB 10968191 IC50 = 22300 nM T07663 C3GAM5 10973079 IC50 = 0.03 nM T07663 C96GWI 10983515 IC50 = 0.7 nM T07663 C84LQY 10983963 Ki = 2.59 nM T07663 CJCO78 10992580 Ki = 1.08 nM T07663 CKX30W 10994934 Ki = 0.61 nM T07663 C3EH8D 11006014 Ki = 24.7 nM T07663 CF7RW4 11016445 Ki = 2.64 nM T07663 CX1GO8 11016581 Ki = 2.71 nM T07663 CR7C1N 11017676 EC50 = 12 nM T07663 CO05WV 11024165 IC50 = 3900 nM T07663 CJMS98 11025421 Ki = 1.2 nM T07663 C3QT7I 11028215 Ki = 0.53 nM T07663 C98IUO 11039211 Ki = 0.76 nM T07663 CF6BL1 11049430 Ki = 62.8 nM T07663 C7B4MG 11071221 Ki = 1.71 nM T07663 CIO28H 11092703 Ki = 0.99 nM T07663 CG74CI 11093245 EC50 = 130 nM T07663 CW2AS4 11103879 Ki = 0.29 nM T07663 CRV32I 11114031 Ki = 3.74 nM T07663 C72TWL 11123617 Ki = 246 nM T07663 CX3N0E 11123630 Ki = 0.31 nM T07663 C24VFA 11125005 EC50 = 37 nM T07663 CL3DT7 11145432 Ki = 0.73 nM T07663 CU5C3E 11145600 Ki = 0.61 nM T07663 C3B1QP 11161553 IC50 = 21000 nM T07663 C6OH2Y 11212743 Ki = 0.22 nM T07663 CA8E0W 11212836 Ki = 0.58 nM T07663 C0FSV9 11225074 IC50 = 0.07 nM T07663 C8TD3U 11247946 IC50 = 0.14 nM T07663 C01VJK 11270159 Ki = 23.3 nM T07663 CF7R3Y 11270592 Ki = 1.06 nM T07663 C26HWL 11270869 IC50 = 0.78 nM T07663 C4R1UG 11270952 Ki = 11 nM T07663 CRZ9V8 11293623 Ki = 3.48 nM T07663 CGO29X 11318932 IC50 = 7600 nM T07663 CY9O2K 11351010 Ki = 0.35 nM T07663 CY71CZ 11351116 Ki = 4.53 nM T07663 C1YTA6 11351932 Ki = 118 nM T07663 CREQ98 11373312 IC50 = 95000 nM T07663 C4H9WX 11375723 IC50 = 320 nM T07663 CVT52P 11385644 Ki = 113 nM T07663 CPJ0Z3 11396900 Ki = 601 nM T07663 C4V6DZ 11418838 Ki = 12.5 nM T07663 C45VZC 11438405 IC50 > 16000 nM T07663 CKZ43J 11496164 IC50 = 0.08 nM T07663 CO9WX8 11497051 IC50 = 1.7 nM T07663 CS5P1N 11502459 IC50 = 2.1 nM T07663 C7S4QZ 11539946 IC50 = 1.01 nM T07663 C4ZYH9 11547485 IC50 = 2.5 nM T07663 C50BPN 11554196 IC50 = 0.65 nM T07663 CJ41RB 11560313 IC50 = 0.4 nM T07663 CJ1R6X 11568346 IC50 = 0.007 nM T07663 CL83VR 11574797 IC50 = 0.65 nM T07663 C86YZS 11575452 IC50 = 0.78 nM T07663 C53ARX 11582654 IC50 = 9.52 nM T07663 C1TOQ3 11583812 IC50 = 6.48 nM T07663 CY5JK4 11589901 IC50 = 34 nM T07663 CI6AW2 11590842 IC50 = 0.09 nM T07663 C58OXQ 11596704 IC50 = 3.3 nM T07663 CG5LT6 11605112 IC50 = 3.15 nM T07663 C7JLT3 11611915 IC50 = 0.07 nM T07663 CLU3G9 11639525 IC50 = 10 nM T07663 CO6XA4 11647832 IC50 = 0.72 nM T07663 CRK10B 11669288 IC50 = 67 nM T07663 C0B7RV 11675647 IC50 = 1.5 nM T07663 C1WV4T 11682414 IC50 = 0.5 nM T07663 C5LPU2 11690391 IC50 = 0.76 nM T07663 C5PHZ0 11710213 IC50 = 1300 nM T07663 CT69CO 11718514 IC50 = 2.6 nM T07663 C1RX0I 11720166 IC50 = 0.35 nM T07663 C7BAC0 11724504 IC50 = 4300 nM T07663 CM5T9U 11724564 IC50 = 35000 nM T07663 CNL0G1 11725859 IC50 = 10 nM T07663 C0AKJ4 11742456 IC50 > 100000 nM T07663 CA1E6R 11754694 Ki = 0.53 nM T07663 C26CKE 11754697 IC50 = 300 nM T07663 C6ERQ9 11755313 Ki = 18 nM T07663 CMP35Y 11762536 Ki = 0.15 nM T07663 C57BPZ 11763070 Ki = 1.3 nM T07663 C1K3JX 11764545 IC50 = 37000 nM T07663 CF23VJ 11775013 IC50 = 0.5012 nM T07663 C23DSJ 11782534 IC50 = 9300 nM T07663 C5EFC7 11793221 IC50 = 1000 nM T07663 CGA1F8 11794425 IC50 = 3000 nM T07663 CUM8A9 11795949 IC50 = 4300 nM T07663 C3LO2Q 11799196 IC50 = 3.1 nM T07663 C0GP6R 11812647 Ki = 0.35 nM T07663 C1J9UP 11813138 Ki = 0.52 nM T07663 CMU6W8 11826705 Ki = 1.74 nM T07663 CB4RS5 11826881 Ki = 2.09 nM T07663 C29HOL 11828590 EC50 = 44 nM T07663 CT5C0K 11849942 IC50 = 100 nM T07663 CS42FO 11849943 IC50 = 240 nM T07663 C2FZY3 11850012 IC50 = 470 nM T07663 CRY1U7 11850013 IC50 = 140 nM T07663 CVJ1X4 11850014 IC50 = 50 nM T07663 CAPF41 11850015 IC50 = 180 nM T07663 C4GQ2P 11850016 IC50 = 38 nM T07663 C4YP5D 11850079 IC50 = 40 nM T07663 C8VUW0 11850080 IC50 = 23 nM T07663 CJ6ZX9 11850081 IC50 = 8.3 nM T07663 CQ2JU9 11850082 IC50 = 79 nM T07663 CSI25Y 11850083 IC50 = 95 nM T07663 CW6D5J 11850144 IC50 = 370 nM T07663 CT9LD7 11850145 IC50 = 1500 nM T07663 C14ZXU 11850147 IC50 = 390 nM T07663 CU7X9W 11850294 IC50 = 71 nM T07663 C8ZM2F 11850366 IC50 = 220 nM T07663 CLI6G9 11850367 IC50 = 100 nM T07663 CC59AF 11850439 IC50 = 1400 nM T07663 CUK49V 11988837 Ki = 600 nM T07663 CFIO49 11988967 Ki = 1600 nM T07663 C2D0NG 11989101 Ki = 590 nM T07663 C65ABT 11989102 Ki = 1200 nM T07663 C05CLB 11992443 IC50 = 0.68 nM T07663 C0Z3KV 11992527 IC50 = 0.9 nM T07663 CXW57M 11992528 IC50 = 0.26 nM T07663 CH86SQ 11992529 IC50 = 0.11 nM T07663 CIX0V4 11992531 IC50 = 1.05 nM T07663 C7X4LC 11992631 IC50 = 0.78 nM T07663 C1B4XD 11992634 IC50 = 0.05 nM T07663 CAG1U6 11992635 IC50 = 0.1 nM T07663 CHT82G 11992739 IC50 = 0.09 nM T07663 CR4CA6 11992740 IC50 = 0.14 nM T07663 CIOU94 11992741 IC50 = 0.25 nM T07663 C95DJC 11992742 IC50 = 0.24 nM T07663 C0KM5I 11992827 IC50 = 1.1 nM T07663 CM57ID 11992831 IC50 = 0.07 nM T07663 CPX16N 11993169 IC50 = 0.07 nM T07663 C0Q4KT 11993170 IC50 = 0.04 nM T07663 C3HOV8 11993171 IC50 = 0.05 nM T07663 CZ7YR6 11993243 IC50 = 2.59 nM T07663 C4VY3X 11993244 IC50 = 0.34 nM T07663 CP4J1S 11993342 IC50 = 0.14 nM T07663 C0QZ6W 11993365 IC50 = 0.15 nM T07663 COQ5N2 11993435 IC50 = 0.43 nM T07663 C39KLP 11993437 IC50 = 1.17 nM T07663 CL8TM7 11993463 IC50 = 0.13 nM T07663 C1ZDC4 11993465 IC50 = 0.08 nM T07663 CK63SM 11993560 IC50 = 1.65 nM T07663 CIRM68 11993561 IC50 = 0.07 nM T07663 C6W2LU 11993562 IC50 = 0.13 nM T07663 C6VI5Z 12020635 Ki = 126 nM T07663 C48IYW 12020642 Ki = 24 nM T07663 CJC01W 12020645 Ki > 1000 nM T07663 CJ4H1G 12020670 Ki = 123 nM T07663 C6D0MG 12069381 IC50 = 1.4 nM T07663 C6S8LD 12355883 IC50 = 1500 nM T07663 CX0C7I 12993019 Ki = 543 nM T07663 CNR05L 12993020 Ki = 126 nM T07663 CO3G0B 12993027 Ki = 0.98 nM T07663 C09OJP 12993038 Ki = 2.07 nM T07663 CI18JL 13026433 IC50 = 1610 nM T07663 C51CKG 14583584 IC50 = 45500 nM T07663 C2ZX8H 14756622 IC50 = 1000 nM T07663 CVT43Z 15473392 IC50 = 60 nM T07663 C2RT6A 15500912 IC50 = 1.9 nM T07663 C8E4IH 15524307 IC50 = 11 nM T07663 C12BUL 15524308 IC50 = 19 nM T07663 CAC5H0 15606258 IC50 = 91000 nM T07663 C3BI9R 15951010 IC50 > 2000 nM T07663 CW6MV8 15981426 IC50 = 26 nM T07663 CYE3L9 16038477 IC50 = 2.6 nM T07663 C9OF5R 16038616 IC50 = 3.7 nM T07663 C8FJM7 16038617 IC50 = 4.5 nM T07663 C4T6CP 16038618 IC50 = 1.2 nM T07663 CIR42U 16038756 IC50 = 12 nM T07663 CF3UG1 16066664 IC50 = 0.04 nM T07663 CG1V8D 17799315 IC50 = 2.7 nM T07663 C1PZ8C 18734933 IC50 > 16000 nM T07663 C6OJI9 18796635 IC50 = 8900 nM T07663 C1FJL6 18796640 IC50 > 100000 nM T07663 CRJO82 18796649 IC50 = 4000 nM T07663 CA16YO 18796653 IC50 = 780 nM T07663 CKCM70 18796657 IC50 = 2200 nM T07663 C36LEN 18796668 IC50 = 1300 nM T07663 C0L8NR 18796689 IC50 = 1900 nM T07663 CBF8M6 18796697 IC50 = 1000 nM T07663 C3RH7V 18796719 IC50 = 11000 nM T07663 CC2WD9 18796725 IC50 > 100000 nM T07663 CNSH93 18796735 IC50 = 2000 nM T07663 CHK4Z7 18796752 IC50 = 32000 nM T07663 CNZ3I1 18796756 IC50 = 4600 nM T07663 CC1LP2 18796767 IC50 = 1000 nM T07663 C2FN9A 18796769 IC50 = 26000 nM T07663 CUE4A2 18796773 IC50 = 2000 nM T07663 C02JXD 18796791 IC50 = 1700 nM T07663 CQ8I5K 18796795 IC50 = 3500 nM T07663 CDC76R 20299686 IC50 = 26 nM T07663 CNX2D5 20646826 IC50 = 0.86 nM T07663 C36XCM 20646828 IC50 = 4.4 nM T07663 C1H2WT 20709323 IC50 = 1.8 nM T07663 C58VPG 21212519 IC50 = 2100 nM T07663 CXM8E3 21704212 IC50 = 0.79 nM T07663 CRY9Z1 21704213 IC50 = 0.32 nM T07663 CS09OZ 21704217 IC50 = 0.5 nM T07663 CH53WM 21704221 IC50 = 14 nM T07663 C7RK1W 21920272 IC50 = 5180 nM T07663 CH7N9S 21920275 IC50 = 7000 nM T07663 CV04DH 21920370 IC50 > 101000 nM T07663 C97JPF 22004355 IC50 = 6.7 nM T07663 C7DJ9E 22004357 IC50 = 2.6 nM T07663 CY6QT7 22004369 IC50 = 1.7 nM T07663 C2STP3 22004386 IC50 = 6.8 nM T07663 C7ZH2R 22004388 IC50 = 0.3 nM T07663 COM30K 22004392 IC50 = 0.7 nM T07663 C37JNS 22004412 IC50 = 0.7 nM T07663 C64YFT 22226537 IC50 = 553 nM T07663 C5G6BS 22226562 IC50 = 30 nM T07663 C70JWO 22226563 IC50 = 94 nM T07663 C8TEV5 22601583 IC50 = 0.4 nM T07663 C2FMU0 22601651 IC50 = 1.3 nM T07663 CNGD52 22744443 IC50 = 1.2 nM T07663 CMIO49 23527107 IC50 = 100 nM T07663 CZD94A 23527108 IC50 = 19 nM T07663 CW96SI 23624262 IC50 = 561 nM T07663 CXB78L 23624298 IC50 > 5000 nM T07663 C4S6VD 23654252 IC50 > 50000 nM T07663 CAJ57O 24751843 IC50 = 79000 nM T07663 CR0D6X 24751988 IC50 > 400000 nM T07663 CL79TD 24751991 IC50 = 65000 nM T07663 C51ZNR 24774842 IC50 > 5000 nM T07663 CQ19ZC 24775191 IC50 = 3500 nM T07663 C9WGI4 24802717 IC50 = 919 nM T07663 C4Y3FK 24883368 IC50 = 1.6 nM T07663 C5F6SD 24956185 IC50 = 26 nM T07663 CA9PN0 24957913 IC50 = 17 nM T07663 C6EQG2 24963293 IC50 = 0.2 nM T07663 CJ43BX 24963638 IC50 = 0.18 nM T07663 CLDO78 24963639 IC50 = 0.72 nM T07663 CG1BJ3 24965774 IC50 = 0.21 nM T07663 CDC01R 24965775 IC50 = 0.33 nM T07663 CDF34R 24966125 IC50 = 0.22 nM T07663 CNO40A 24966126 IC50 = 0.3 nM T07663 CY0G1A 24966127 IC50 = 0.23 nM T07663 CS56UN 24966128 IC50 = 1.08 nM T07663 CA25UL 24969619 IC50 = 0.31 nM T07663 C3AFU0 25093775 IC50 = 3.28 nM T07663 C93DZI 25147798 IC50 > 50000 nM T07663 CPC08B 25179287 IC50 > 50000 nM T07663 COB03R 25179478 IC50 = 40000 nM T07663 C1AV7L 30105766 IC50 = 8 nM T07663 C43UKE 42628078 IC50 = 2.4 nM T07663 CICF39 42629702 IC50 = 1850 nM T07663 CM3X9S 42629827 IC50 > 1000 nM T07663 CQN26J 42629945 IC50 = 1240 nM T07663 C6O5FX 42630062 IC50 = 2080 nM T07663 C71ZNR 42630180 IC50 = 1440 nM T07663 C4RHY0 42630191 IC50 > 5000 nM T07663 CT6RS9 42630192 IC50 = 5165 nM T07663 CYZL43 42630317 IC50 = 8780 nM T07663 CH42OZ 42630318 IC50 > 5000 nM T07663 C7X5AH 42630437 IC50 = 2050 nM T07663 CEPY38 43826154 IC50 = 200000 nM T07663 CQU19I 44180409 IC50 = 30300 nM T07663 CW8OB3 44243146 Ki = 10600 nM T07663 C19SIQ 44249786 IC50 = 14.5 nM T07663 C03DAV 44249787 IC50 = 2.3 nM T07663 CJ1GS3 44249944 IC50 = 0.9 nM T07663 CAL8X3 44264943 IC50 = 1 nM T07663 C59QCJ 44274690 IC50 = 3.89 nM T07663 C9KV6Y 44274762 IC50 = 6.457 nM T07663 CXA6Y3 44274773 IC50 = 0.61 nM T07663 CF4H9A 44274775 IC50 = 0.8913 nM T07663 CW7J4K 44274797 IC50 = 1.995 nM T07663 C9VK6M 44274798 IC50 = 5.012 nM T07663 CTP4O5 44274817 IC50 = 2.818 nM T07663 CA6J8T 44274920 IC50 = 3000 nM T07663 CV1ZA7 44280486 IC50 = 3.6 nM T07663 CG8R0W 44280487 IC50 = 4 nM T07663 CS0FX4 44280546 IC50 = 2.7 nM T07663 C05SIA 44280556 IC50 = 12.8 nM T07663 CA9KV4 44280558 IC50 = 8.4 nM T07663 CY74KE 44280614 IC50 = 19.8 nM T07663 C4RO9D 44280635 IC50 = 2.5 nM T07663 CH7W2T 44280722 IC50 = 1.2 nM T07663 CTO54N 44280723 IC50 = 0.7 nM T07663 CXRU70 44280792 IC50 = 13.2 nM T07663 CO7NV0 44280794 IC50 = 164 nM T07663 CG8I6M 44280801 IC50 = 57 nM T07663 CDQ8B2 44280847 IC50 = 1.5 nM T07663 C0N3JE 44280911 IC50 = 2 nM T07663 C3DHJ2 44280985 IC50 = 1.9 nM T07663 CA3GF6 44280994 IC50 = 127 nM T07663 CXB40D 44281036 IC50 = 28.6 nM T07663 CA1HN8 44281061 IC50 = 15.7 nM T07663 C7TKW4 44281095 IC50 = 7.1 nM T07663 CK3W1B 44281096 IC50 = 4 nM T07663 CC81DV 44281265 IC50 = 132 nM T07663 CNO94A 44281273 IC50 > 1000 nM T07663 CO1L0H 44282267 IC50 = 160 nM T07663 C79RGL 44282685 IC50 = 270 nM T07663 CK8Y4F 44286951 IC50 = 160 nM T07663 CNW8B7 44287071 IC50 = 73 nM T07663 CDHP47 44287318 IC50 = 0.6 nM T07663 C2O0JN 44307127 IC50 = 530 nM T07663 C2FW1A 44310350 IC50 = 2900 nM T07663 COP54Y 44318505 IC50 = 1.5 nM T07663 CK0N6P 44318516 IC50 = 0.95 nM T07663 C4AWN5 44318518 IC50 = 1.23 nM T07663 CP30VE 44318806 IC50 = 0.73 nM T07663 CH4T3J 44318846 IC50 = 0.7 nM T07663 CKLM51 44318862 IC50 = 150 nM T07663 CX5SO4 44320719 IC50 = 77 nM T07663 C1SI7O 44320739 IC50 = 551 nM T07663 C3TZ6O 44320740 IC50 = 105 nM T07663 CH18VT 44320762 IC50 = 135 nM T07663 C45ZJD 44320781 IC50 = 130 nM T07663 CF1DO2 44320804 IC50 = 160 nM T07663 CLBV45 44320831 IC50 = 28 nM T07663 C6RS5T 44320847 IC50 = 1360 nM T07663 CVS5D1 44320863 IC50 = 20 nM T07663 C0GM7F 44320900 IC50 = 315 nM T07663 C13WMT 44320988 IC50 = 12 nM T07663 CP78QN 44320989 IC50 = 26 nM T07663 CP34EA 44321012 IC50 = 63 nM T07663 CN8Z1I 44321013 IC50 = 24 nM T07663 CDP87G 44321026 IC50 = 3.5 nM T07663 C9G0OQ 44321064 IC50 = 19 nM T07663 CWMD23 44321111 IC50 = 5.5 nM T07663 CPEB60 44321112 IC50 = 10 nM T07663 CX9L7V 44321135 IC50 = 11 nM T07663 C51CET 44321137 IC50 = 5 nM T07663 CD0QO6 44321152 IC50 = 93 nM T07663 C69MZC 44321154 IC50 = 5420 nM T07663 CUV0W1 44321156 IC50 > 10000 nM T07663 CP71YV 44321172 IC50 = 16 nM T07663 CXNO48 44321173 IC50 > 10000 nM T07663 C7NE6Q 44321175 IC50 > 10000 nM T07663 C81WUS 44321176 IC50 = 1500 nM T07663 C4QO0A 44321178 IC50 > 10000 nM T07663 CZWA59 44321202 IC50 = 60 nM T07663 C4B1WH 44321204 IC50 = 73 nM T07663 CIAN09 44321224 IC50 = 1810 nM T07663 C86ATM 44321229 IC50 = 100 nM T07663 CR54IA 44321231 IC50 > 10000 nM T07663 C4VFQ5 44321253 IC50 = 91 nM T07663 CYVA51 44321254 IC50 > 10000 nM T07663 CUQ3R1 44321255 IC50 = 100 nM T07663 C7BM6I 44321261 IC50 = 59 nM T07663 CZ16IY 44324251 IC50 = 30000 nM T07663 CCX9Z3 44324252 IC50 = 24000 nM T07663 CG6UT1 44324296 IC50 = 20000 nM T07663 C8M4WJ 44324373 IC50 = 22000 nM T07663 CY5HZ7 44324390 IC50 = 9000 nM T07663 C5KYV6 44324391 IC50 = 8000 nM T07663 C5C4QX 44324507 IC50 = 22000 nM T07663 CNK2F8 44331802 IC50 = 270 nM T07663 CGFP09 44336826 IC50 = 0.82 nM T07663 C98VIX 44336827 IC50 = 0.69 nM T07663 C1L6SG 44336834 IC50 = 1.1 nM T07663 CH8RY1 44336844 IC50 = 1.8 nM T07663 C1AC3Z 44336847 IC50 = 0.3 nM T07663 C0NT4K 44336855 IC50 = 0.33 nM T07663 C9WLD8 44336856 IC50 = 2 nM T07663 CUME98 44336924 IC50 = 0.58 nM T07663 CM1BO3 44348247 IC50 = 32000 nM T07663 CY5L6J 44348257 IC50 = 11000 nM T07663 CD5ZW3 44348484 IC50 = 650 nM T07663 C80PGJ 44348564 IC50 = 1500 nM T07663 CY0T1M 44348625 IC50 = 9600 nM T07663 CG98RE 44358477 Ki = 3.32 nM T07663 C3H4MR 44358478 Ki = 2.49 nM T07663 CBD52Z 44358886 Ki = 4.66 nM T07663 C7LN0W 44363056 IC50 = 50 nM T07663 C71YUD 44363183 IC50 = 3000 nM T07663 CF0IB6 44377834 IC50 = 105 nM T07663 CWO45S 44377842 Ki = 145 nM T07663 C27ZVC 44377867 Ki = 132 nM T07663 C7TXQ3 44377869 Ki = 179 nM T07663 CSW1J4 44377881 Ki = 219 nM T07663 C27TDG 44377933 Ki > 100 nM T07663 C8XM3I 44377988 IC50 = 100 nM T07663 C5IOH4 44378004 IC50 = 95 nM T07663 C85XCK 44378015 Ki = 850 nM T07663 C0H7KF 44378030 Ki > 5000 nM T07663 CU29OZ 44378056 Ki = 130 nM T07663 CLV13K 44378110 Ki > 10000 nM T07663 CL3SI5 44378121 Ki = 50.6 nM T07663 CYA76O 44378142 IC50 > 10000 nM T07663 C6IOU8 44378149 Ki = 8.11 nM T07663 CBQ5W3 44378155 IC50 = 67 nM T07663 CR30BD 44378165 Ki = 32.3 nM T07663 CHL5D9 44378187 Ki = 77.5 nM T07663 CV5Y1A 44378199 Ki = 64.2 nM T07663 CT8NH9 44383851 IC50 > 10000 nM T07663 C19CRH 44383901 IC50 = 19700 nM T07663 CR9O3I 44383902 IC50 > 30000 nM T07663 CW47HV 44383906 IC50 = 17700 nM T07663 CL86MY 44383907 IC50 > 10000 nM T07663 CW63HQ 44383912 IC50 > 10000 nM T07663 CF98LG 44384286 IC50 > 10000 nM T07663 CN1WS7 44384345 IC50 = 66700 nM T07663 C01XPL 44384404 IC50 = 22700 nM T07663 CWPR87 44384405 IC50 = 2900 nM T07663 C59SDR 44384406 IC50 = 3900 nM T07663 C7WT4G 44384540 IC50 = 18200 nM T07663 C4RQB0 44384541 IC50 = 21200 nM T07663 CRZ5G8 44384546 IC50 > 100000 nM T07663 C6W4GY 44384713 IC50 = 56100 nM T07663 CKH7M8 44384714 IC50 > 30000 nM T07663 C0ZGU6 44385109 IC50 = 12100 nM T07663 CE80VB 44385244 IC50 = 1700 nM T07663 CH5GU8 44385282 IC50 = 14900 nM T07663 CL50UE 44385283 IC50 = 9700 nM T07663 CSN56E 44386916 IC50 = 3.981 nM T07663 C13HPW 44393651 IC50 > 101000 nM T07663 CJ6GB5 44393709 IC50 = 11600 nM T07663 CQP01D 44393950 IC50 = 18770 nM T07663 CU1CQ8 44394047 IC50 = 80000 nM T07663 CJYC83 44397324 IC50 = 2070 nM T07663 CZUY06 44397327 IC50 = 5620 nM T07663 CB64FY 44397328 IC50 = 1690 nM T07663 CDJ87T 44397345 IC50 = 6190 nM T07663 C5CTF6 44397346 IC50 = 140 nM T07663 C2T7BQ 44397347 IC50 = 680 nM T07663 C39VBJ 44397348 IC50 = 3350 nM T07663 CU3BF4 44397365 IC50 = 1840 nM T07663 CRTY10 44397366 IC50 = 2930 nM T07663 CYFD01 44397379 IC50 = 1510 nM T07663 C4VS1H 44397382 IC50 = 74 nM T07663 C8YCU6 44397384 IC50 = 3190 nM T07663 CQD8Z7 44397386 IC50 = 13 nM T07663 CCL9D6 44397387 IC50 = 620 nM T07663 CSAQ43 44397397 IC50 = 3190 nM T07663 C7MZ8J 44397413 IC50 = 5990 nM T07663 C8KA6R 44397415 IC50 = 920 nM T07663 CR8P4T 44397447 IC50 = 3280 nM T07663 C9TK8I 44397448 IC50 = 5150 nM T07663 CF2AP3 44397474 IC50 = 230 nM T07663 CQT12O 44397490 IC50 = 2720 nM T07663 C6FJV7 44397494 IC50 = 1280 nM T07663 CZ5QV6 44397495 IC50 = 2130 nM T07663 CAP7W0 44397504 IC50 = 1210 nM T07663 CU13ES 44397515 IC50 = 96 nM T07663 CQY79V 44397539 IC50 = 8900 nM T07663 CTAI27 44397548 IC50 = 1470 nM T07663 C98ZCS 44397556 IC50 = 270 nM T07663 CMC12S 44397573 IC50 = 6490 nM T07663 CL15YW 44397574 IC50 = 3810 nM T07663 C6GIS2 44397576 IC50 = 10000 nM T07663 C65PLD 44397577 IC50 = 4520 nM T07663 C8MFC2 44397582 IC50 = 3300 nM T07663 C3PN4D 44397598 IC50 = 790 nM T07663 CE2GZ3 44397599 IC50 = 6680 nM T07663 CY0KB5 44397600 IC50 = 2660 nM T07663 C86IAQ 44397602 IC50 = 1900 nM T07663 CR0D6I 44397603 IC50 = 8760 nM T07663 CD67XW 44397612 IC50 = 6090 nM T07663 C1ISA5 44397619 IC50 = 7820 nM T07663 CG2XI7 44397621 IC50 = 6250 nM T07663 C1HBU8 44397622 IC50 = 3160 nM T07663 CA1FG3 44397627 IC50 = 9070 nM T07663 C1FJH9 44397640 IC50 = 74 nM T07663 CV2Q1K 44397643 IC50 = 17 nM T07663 C69WZC 44397646 IC50 = 130 nM T07663 CC8Z3A 44397647 IC50 = 3680 nM T07663 C1VB8P 44397694 IC50 = 630 nM T07663 CV2M0A 44397708 IC50 = 3500 nM T07663 C8MZF1 44397709 IC50 = 4580 nM T07663 C2OA3Y 44397724 IC50 = 9460 nM T07663 CJIK26 44397727 IC50 = 320 nM T07663 CFP7S8 44397728 IC50 = 350 nM T07663 CERQ57 44397746 IC50 = 2640 nM T07663 C2PJ6R 44397748 IC50 = 10000 nM T07663 CAQD83 44397749 IC50 = 1100 nM T07663 C5GLC2 44397761 IC50 = 40 nM T07663 CUZY95 44397764 IC50 = 8620 nM T07663 CQCN29 44397781 IC50 = 770 nM T07663 C0B2YM 44397782 IC50 = 830 nM T07663 CWL0A9 44397785 IC50 = 3410 nM T07663 CSN79W 44397799 IC50 = 1800 nM T07663 C20BLM 44397801 IC50 = 1830 nM T07663 CJG87Q 44397802 IC50 = 500 nM T07663 CP1CU7 44397810 IC50 = 650 nM T07663 CI7HS1 44397811 IC50 = 6070 nM T07663 C9SQ1V 44397814 IC50 = 1450 nM T07663 CZF29N 44397816 IC50 = 190 nM T07663 CIVF18 44397836 IC50 = 890 nM T07663 CP18FI 44397837 IC50 = 2580 nM T07663 CRMN86 44397859 IC50 = 3200 nM T07663 CC7B3S 44397860 IC50 = 460 nM T07663 C01CAI 44397871 IC50 = 10000 nM T07663 C8Y0WF 44397874 IC50 = 7650 nM T07663 CJ6B1W 44397876 IC50 = 2420 nM T07663 C28ERI 44397877 IC50 = 2490 nM T07663 C6Y9XN 44397888 IC50 = 520 nM T07663 CIOM21 44397889 IC50 = 430 nM T07663 CVQ8C1 44397891 IC50 = 1240 nM T07663 CX3M5J 44397892 IC50 = 270 nM T07663 CYX72U 44397904 IC50 = 3100 nM T07663 C5JS4T 44397906 IC50 = 8910 nM T07663 CVB7K2 44397908 IC50 = 2200 nM T07663 CP8CW5 44397940 IC50 = 9430 nM T07663 CFHR09 44397941 IC50 = 9280 nM T07663 CP62TK 44397956 IC50 = 4990 nM T07663 C6UY9Z 44397957 IC50 = 4250 nM T07663 C23GTH 44397958 IC50 = 8430 nM T07663 CG36QI 44397976 IC50 = 10000 nM T07663 CDK84C 44397977 IC50 = 7560 nM T07663 CB3ZG1 44397979 IC50 = 1030 nM T07663 C4AO1D 44397980 IC50 = 9870 nM T07663 CW65CR 44397987 IC50 = 5470 nM T07663 C1DQW5 44397991 IC50 = 40 nM T07663 CP8F9A 44397992 IC50 = 8580 nM T07663 CM1ZW4 44401687 IC50 = 230 nM T07663 C0YZV7 44401690 IC50 = 33 nM T07663 C7CDY2 44401692 IC50 = 74 nM T07663 CT8R0Q 44401694 IC50 = 81 nM T07663 CDSE04 44401695 IC50 = 90 nM T07663 CB3RC6 44401705 IC50 = 60 nM T07663 CA59PR 44401708 IC50 = 81 nM T07663 CXA4D6 44401724 IC50 = 23 nM T07663 C17ODM 44401727 IC50 = 430 nM T07663 CX0AZ7 44401742 IC50 = 270 nM T07663 C3G2RU 44401767 IC50 = 350 nM T07663 C4BJ3U 44401771 IC50 = 38 nM T07663 C0F9ZD 44401772 IC50 = 2.3 nM T07663 CM45YT 44401790 IC50 = 33 nM T07663 CA1SR3 44401812 IC50 = 29 nM T07663 CN63AH 44401816 IC50 = 30 nM T07663 CVOW53 44401827 IC50 = 32 nM T07663 CVCN36 44401831 IC50 = 920 nM T07663 C59TYU 44401851 IC50 = 200 nM T07663 C78VHO 44401870 IC50 = 13000 nM T07663 CSM4X8 44401879 IC50 = 20 nM T07663 CZU4T7 44401880 IC50 = 3.3 nM T07663 C01BEI 44401886 IC50 = 100 nM T07663 CU4AR1 44401892 IC50 = 5.3 nM T07663 C14LNK 44401904 IC50 = 60 nM T07663 CVPZ92 44401905 IC50 = 28 nM T07663 C0BRH8 44401908 IC50 = 450 nM T07663 CN4T6Z 44401928 IC50 = 145 nM T07663 CV17OM 44401929 IC50 = 14 nM T07663 CK9VN7 44401931 IC50 = 320 nM T07663 C9Q1ET 44401943 IC50 = 40 nM T07663 CB98IX 44401972 IC50 = 130 nM T07663 CD51UN 44401977 IC50 = 100 nM T07663 C19QCE 44401981 IC50 = 48 nM T07663 C04BTX 44401982 IC50 = 15 nM T07663 C7MY1S 44402027 IC50 = 59 nM T07663 C6XA7P 44402060 IC50 = 3100 nM T07663 CTZ52C 44402073 IC50 = 28 nM T07663 C4P8RN 44402077 IC50 = 35 nM T07663 C6S8KA 44402114 IC50 = 40 nM T07663 CDNZ52 44402130 IC50 = 180 nM T07663 CP78NL 44402133 IC50 = 1100 nM T07663 CWVH96 44402149 IC50 = 100 nM T07663 C9BN6H 44402168 IC50 = 6.5 nM T07663 CQM65U 44402195 IC50 = 160 nM T07663 CM90NL 44402196 IC50 = 980 nM T07663 C6IY5O 44402213 IC50 = 39 nM T07663 C4O7QE 44402239 IC50 = 22 nM T07663 C4P0AC 44402278 IC50 = 75 nM T07663 C1GPC2 44402295 IC50 = 7.8 nM T07663 CCZ2E8 44438552 IC50 = 462 nM T07663 CB1C2M 44438553 IC50 = 25 nM T07663 C7RV5Q 44438554 IC50 = 20 nM T07663 CCOJ06 44438555 IC50 = 28 nM T07663 CB93RX 44438557 IC50 = 33 nM T07663 C9AO2Z 44438558 IC50 = 42 nM T07663 C50ZMB 44438560 IC50 = 5 nM T07663 C39ZMJ 44438561 IC50 = 26 nM T07663 CBQN25 44438563 IC50 = 10000 nM T07663 CJH70L 44438564 IC50 = 34 nM T07663 CE4S8J 44438565 IC50 = 51 nM T07663 CK1JU3 44459193 IC50 = 1.288 nM T07663 CZFU59 44459332 IC50 = 43 nM T07663 CJ0Q4D 44459333 IC50 = 2.2 nM T07663 CT39RH 44459469 IC50 = 2.8 nM T07663 CG4AI3 44459482 IC50 = 2.089 nM T07663 CZ6IU2 44459494 IC50 = 6.457 nM T07663 C68RBI 44459495 IC50 = 5.37 nM T07663 CNJ16Q 44459505 IC50 = 4.5 nM T07663 C0FQ1O 44459535 IC50 = 5 nM T07663 CT9R7K 44459542 IC50 = 46 nM T07663 CP97OV 44459564 IC50 = 57.54 nM T07663 C49NWP 44459572 IC50 = 550 nM T07663 C5G2JO 44459598 IC50 = 19.95 nM T07663 C8MBD9 44459599 IC50 = 158.49 nM T07663 C0W4VT 44459622 IC50 = 39.81 nM T07663 C18EJF 44459640 IC50 = 1.8 nM T07663 C7RGD3 44459641 IC50 = 2.089 nM T07663 CQ95TO 44459661 IC50 = 128.82 nM T07663 CRH7N1 44459687 IC50 = 6.31 nM T07663 C8JS2X 44459694 IC50 = 18 nM T07663 CO3F9K 44459713 IC50 = 8.3 nM T07663 CF4C3P 44459717 IC50 = 7 nM T07663 C1W5OG 44459718 IC50 = 21.88 nM T07663 C31SQM 44459720 IC50 = 2.291 nM T07663 CS17XE 44459751 IC50 = 6.761 nM T07663 C85QDR 44459752 IC50 = 13 nM T07663 CI2V6T 44459760 IC50 = 1.096 nM T07663 CJN91Z 44459761 IC50 = 0.8913 nM T07663 CQ01TE 44459776 IC50 = 3.09 nM T07663 C24BGR 44459782 IC50 = 1.514 nM T07663 CB37LV 44459783 IC50 = 6.3 nM T07663 C1V3CW 44459848 IC50 = 3.02 nM T07663 C52JOE 44459875 IC50 = 47.86 nM T07663 CZ1DJ8 44459876 IC50 = 55 nM T07663 CWXV09 44459906 IC50 = 0.3 nM T07663 CJ4L3O 44459907 IC50 = 7.943 nM T07663 CZ0DN5 44572149 IC50 > 10000 nM T07663 C6U8QW 44572150 IC50 > 10000 nM T07663 C9XD8C 44572789 IC50 = 5200 nM T07663 C72XEI 44572984 IC50 > 10000 nM T07663 CIX5Q0 44572985 IC50 > 10000 nM T07663 C7UXN8 44572986 IC50 > 10000 nM T07663 CRBQ49 44572987 IC50 = 6500 nM T07663 C0WXB4 44580020 IC50 = 1.585 nM T07663 CHA63L 44580021 IC50 = 6.31 nM T07663 CX3L1P 44587252 IC50 = 160 nM T07663 CI3K8T 44605342 IC50 = 87100 nM T07663 CV8RY3 45260952 IC50 = 3 nM T07663 CLEU14 45260983 IC50 = 12 nM T07663 C48QSY 45261659 IC50 = 1700 nM T07663 CC5Z7N 45261660 IC50 = 2300 nM T07663 C26IBG 45261674 IC50 = 5000 nM T07663 CTG0D9 45261728 IC50 = 2800 nM T07663 CS7GA3 45264997 IC50 = 760 nM T07663 C3IOB7 45265000 IC50 = 360 nM T07663 CKW39R 45267744 IC50 = 4.571 nM T07663 C9PC5S 45267756 IC50 = 223.87 nM T07663 CR7QN3 45267764 IC50 = 0.3 nM T07663 C1KTZ3 45267771 IC50 = 33.9 nM T07663 C6WLB4 45268626 IC50 = 2.5 nM T07663 CE0U3W 45268639 IC50 = 13.49 nM T07663 CR8JH9 45268646 IC50 = 33.3 nM T07663 CM8OP3 45268652 IC50 = 0.3 nM T07663 CD6A0O 45269469 IC50 = 20.3 nM T07663 CL42XG 45269481 IC50 = 3.467 nM T07663 CRWE76 45269493 IC50 = 0.4 nM T07663 CHN4F0 45269499 IC50 = 2.9 nM T07663 C6DQU1 45269515 IC50 = 534 nM T07663 CB4IO3 45269516 IC50 = 51 nM T07663 CD47UP 45270308 IC50 = 28.18 nM T07663 C4VPC6 45270320 IC50 = 1 nM T07663 CMF3T7 45270338 IC50 = 36.5 nM T07663 C1XZ4Q 45270704 IC50 = 1.21 nM T07663 C89NBL 45270705 IC50 = 1.21 nM T07663 CDWX76 45271142 IC50 = 147.91 nM T07663 C62LVH 45272043 IC50 = 52.5 nM T07663 C0AO8K 45272078 IC50 = 43 nM T07663 CN7GR1 45272848 IC50 = 1.995 nM T07663 C8RZ7H 45272849 IC50 = 2.692 nM T07663 CQ34VM 45272857 IC50 = 3 nM T07663 C5H9RX 45272874 IC50 = 22.4 nM T07663 C7X2VE 45272888 IC50 = 0.9 nM T07663 CN8G9K 45272901 IC50 = 26.7 nM T07663 C2MW1C 45272908 IC50 = 25 nM T07663 C3X7RV 45273795 IC50 = 1.288 nM T07663 C74IXB 45273827 IC50 = 0.3 nM T07663 CLZ39M 45379958 IC50 = 2.38 nM T07663 C98KFA 45486490 IC50 = 1.17 nM T07663 CGA65L 45486496 IC50 = 0.17 nM T07663 CZ8JD0 45486497 IC50 = 0.28 nM T07663 CYF73X 45486498 IC50 = 0.38 nM T07663 C86XSZ 45486501 IC50 = 0.55 nM T07663 CDYO49 45486504 IC50 = 0.06 nM T07663 CNW0I9 45486505 IC50 = 0.71 nM T07663 CWQ6Y5 45486511 IC50 = 16.3 nM T07663 CSG37U 45486513 IC50 = 2.59 nM T07663 CEX01M 45486514 IC50 = 0.32 nM T07663 C58IWJ 45486519 IC50 = 0.25 nM T07663 CE3PK0 45486527 IC50 = 0.68 nM T07663 C1ZYT9 45486549 IC50 = 2.95 nM T07663 CHE56F 45486550 IC50 = 0.34 nM T07663 C84NHX 45486564 IC50 = 0.54 nM T07663 CLMZ68 45486571 IC50 = 4 nM T07663 CB2MG1 45486572 IC50 = 0.32 nM T07663 C0MWV4 45486574 IC50 = 0.88 nM T07663 C9SI3E 45486581 IC50 = 0.36 nM T07663 C51CUF 46193118 IC50 = 640 nM T07663 CTP8R1 46193119 IC50 = 38 nM T07663 CDT4U1 46193239 IC50 = 29000 nM T07663 C0W3LE 46193243 IC50 = 100 nM T07663 CKUN01 46193244 IC50 = 88000 nM T07663 CHU8I7 46193370 IC50 = 2800 nM T07663 C7NC9V 46193371 IC50 = 60 nM T07663 CY49DB 46193372 IC50 = 320 nM T07663 CN05XT 46193373 IC50 = 41000 nM T07663 C1Q6WV 46193374 IC50 = 32000 nM T07663 C60KFT 46193375 IC50 = 50 nM T07663 C2J9IH 46193486 IC50 = 260 nM T07663 CJ86KO 46193489 IC50 = 50 nM T07663 CPYK94 46193490 IC50 = 3400 nM T07663 CHUN05 46193595 IC50 = 40 nM T07663 C5IMB2 46239424 Ki = 6400 nM T07663 CKR9P7 46239425 Ki = 8900 nM T07663 C7SLP0 46239531 Ki = 5000 nM T07663 CI1F5C 46239840 Ki > 100000 nM T07663 C26XVS 46240044 Ki = 17324 nM T07663 CC3UF9 46830325 IC50 = 0.15 nM T07663 CE4JU7 46842025 IC50 = 0.27 nM T07663 CR8JC2 46842169 IC50 = 0.27 nM T07663 CF23CG 46842171 IC50 = 0.27 nM T07663 CWY45O 46842322 IC50 = 4.1 nM T07663 CY9UB1 46842324 IC50 = 0.27 nM T07663 CVP3F6 46886964 IC50 = 0.94 nM T07663 CF49HM 46886965 IC50 = 3.92 nM T07663 CQ91ZP 46887034 IC50 = 2.96 nM T07663 CDI09L 46887035 IC50 = 0.38 nM T07663 C8X6IR 46887483 IC50 = 0.3 nM T07663 C51BJT 46887484 IC50 = 0.86 nM T07663 CB3F2M 46887522 IC50 = 1.84 nM T07663 CVX57Z 46887568 IC50 = 3.28 nM T07663 C3GW8T 46887569 IC50 = 9.79 nM T07663 C13VUK 46888519 IC50 = 0.07 nM T07663 C7G5PM 46888541 IC50 = 0.66 nM T07663 C6NIG0 46888542 IC50 = 1.4 nM T07663 CPM4S1 46888559 IC50 = 5.5 nM T07663 CV53IU 46888560 IC50 = 0.89 nM T07663 C9UY1R 46888576 IC50 = 2.5 nM T07663 CE79JU 46888577 IC50 = 1.2 nM T07663 CQ5B2F 46888578 IC50 = 2.3 nM T07663 C8ITU7 46888595 IC50 = 0.2 nM T07663 C0IQ2C 46888596 IC50 = 2 nM T07663 CS6F1J 46888597 IC50 = 0.087 nM T07663 C7B3ZY 46888631 IC50 = 0.42 nM T07663 C8FW5K 46888632 IC50 = 2.3 nM T07663 C57KWS 46888633 IC50 = 0.35 nM T07663 CS27GK 46888659 IC50 = 0.011 nM T07663 C38INP 46888660 IC50 = 0.07 nM T07663 C6WQ5Y 46888661 IC50 = 1.2 nM T07663 CZ3SO4 46888707 IC50 = 0.19 nM T07663 C02RDT 46888708 IC50 = 0.08 nM T07663 CUN72Y 46888738 IC50 = 0.05 nM T07663 C3P2IN 46933992 IC50 = 11000 nM T07663 CHA5Z0 49821469 IC50 > 1000 nM T07663 C1AYP0 49821627 IC50 > 500 nM T07663 C85AXR 49821714 IC50 > 1000 nM T07663 CZS03D 50902030 Ki > 4274 nM T07663 CH2Z1E 50902289 Ki > 7100 nM T07663 C4HJL2 50902291 Ki > 7950 nM T07663 C6A1IU 50902549 Ki > 2000 nM T07663 C3Y2AV 50903255 Ki > 2000 nM T07663 CN41YJ 50925469 IC50 = 2 nM T07663 CQ3RG5 50925470 IC50 = 7 nM T07663 C2E5JK 50940516 IC50 = 850 nM T07663 CEB5T9 50940517 IC50 = 50 nM T07663 C2C0IA 50940656 IC50 = 850 nM T07663 C4I9OJ 50940659 IC50 = 8750 nM T07663 C6F5RK 50940660 IC50 = 300 nM T07663 C9O4LE 50940680 IC50 = 590 nM T07663 CT3H4X 50940682 IC50 = 4140 nM T07663 CN4S0D 50940686 IC50 = 2310 nM T07663 CT8V2L 50940687 IC50 = 12 nM T07663 CP3G6K 50940690 IC50 = 2300 nM T07663 C7MV1Y 50940692 IC50 = 380 nM T07663 CUM0O5 50940699 IC50 = 730 nM T07663 C9IFA6 50940700 IC50 = 50 nM T07663 C7TF6Q 50940701 IC50 = 1200 nM T07663 CI3AG0 50941259 IC50 = 260 nM T07663 CCUK19 50941260 IC50 = 990 nM T07663 CY37HL 50941261 IC50 = 10 nM T07663 CC0QW5 50941262 IC50 = 1340 nM T07663 C5Q9YU 50941264 IC50 = 3300 nM T07663 C7Y8HK 50941365 IC50 = 270 nM T07663 C8WQX5 50941366 IC50 = 1110 nM T07663 C3NK7Q 50941367 IC50 = 4460 nM T07663 C3QEV9 50941368 IC50 = 290 nM T07663 CA3HQ6 50941461 IC50 = 2040 nM T07663 C8LSY4 50941462 IC50 = 190 nM T07663 C4GBV9 50941463 IC50 = 1260 nM T07663 CYL8N5 50941464 IC50 = 1350 nM T07663 C10WDU 50941465 IC50 = 260 nM T07663 C6YM0P 50941551 IC50 = 1270 nM T07663 C6R4YN 50993785 IC50 = 10000 nM T07663 C0M6XL 50993786 IC50 = 10000 nM T07663 C0OR7K 53248667 IC50 > 100000 nM T07663 CS3R1I 53248669 IC50 = 28900 nM T07663 C30RNE 53248670 IC50 = 6400 nM T07663 C1RJ7M 54580520 IC50 > 400000 nM T07663 CCXF36 54580521 IC50 = 145000 nM T07663 CZG36N 54580522 IC50 > 400000 nM T07663 C0NPM8 54580523 IC50 = 225000 nM T07663 C25VSX 54580524 IC50 > 400000 nM T07663 CBT56Y 54581676 IC50 = 5200 nM T07663 C0MN3D 54582527 IC50 = 156000 nM T07663 C6T1QX 54582528 IC50 = 350000 nM T07663 CP4N1Q 54582529 IC50 > 400000 nM T07663 CW1X3G 54583497 IC50 > 400000 nM T07663 CN96IQ 54585432 IC50 > 400000 nM T07663 CH25CO 54586393 IC50 > 400000 nM T07663 C82LED 54586394 IC50 > 400000 nM T07663 CQ1H3C 54587403 IC50 > 400000 nM T07663 C28GAC 54587404 IC50 > 400000 nM T07663 CFX89L 54587804 IC50 = 5700 nM T07663 CGF65A 54670110 IC50 > 30000 nM T07663 C90ZLC 54670399 IC50 > 30000 nM T07663 CLK61N 56587955 IC50 = 0.1 nM T07663 C4TGL7 56648496 IC50 > 1000 nM T07663 CH6C3L 56648679 IC50 > 10000 nM T07663 CCY79V 56648680 IC50 = 3110 nM T07663 CNE96P 56648857 IC50 > 10000 nM T07663 CX86AQ 56648859 IC50 > 1000 nM T07663 CPC3T4 56654131 IC50 > 10000 nM T07663 C0YD3P 56928304 IC50 > 5000 nM T07663 C8RO6A 56929788 IC50 > 1000 nM T07663 CD52CA 57391118 IC50 = 0.02 nM T07663 C7Y4BX 57391119 IC50 = 1.47 nM T07663 C4PSK2 57391120 IC50 = 0.04 nM T07663 CA1TE7 57391121 IC50 = 0.01 nM T07663 CN60KE 57391196 IC50 = 0.09 nM T07663 CM7N8I 57391197 IC50 = 0.05 nM T07663 C7VXN9 57391198 IC50 = 1.3 nM T07663 C7SC4E 57392888 IC50 = 0.44 nM T07663 CG3DF1 57392948 Ki > 10000 nM T07663 CQT1G9 57392966 IC50 = 1.38 nM T07663 CR28IN 57394623 IC50 = 0.38 nM T07663 CHZ67R 57394624 IC50 = 0.27 nM T07663 CE36TV 57394695 Ki = 24400 nM T07663 CLEY35 57396379 IC50 = 0.64 nM T07663 C7W6TP 57396380 IC50 = 0.05 nM T07663 C80CVX 57396381 IC50 = 0.01 nM T07663 C86YCU 57396469 IC50 = 0.1 nM T07663 C3M6EL 57396470 IC50 = 1.64 nM T07663 CPQ91V 57396471 IC50 = 0.22 nM T07663 CP0AB6 57396472 IC50 = 0.28 nM T07663 CNY5Z8 57398261 IC50 = 0.35 nM T07663 CH57NZ 57398879 IC50 = 15.8 nM T07663 CTYR07 57399826 IC50 = 0.04 nM T07663 CL5UP7 57401597 IC50 = 0.36 nM T07663 C37KMA 57401598 IC50 = 0.13 nM T07663 CHQ79W 57401599 IC50 = 0.02 nM T07663 CWG70K 57401600 IC50 = 0.06 nM T07663 CU5KP3 57401601 IC50 = 0.1 nM T07663 C8GD5N 57402376 IC50 = 8.2 nM T07663 CLU6J0 57403348 IC50 = 2.43 nM T07663 CD73NJ 57403349 IC50 = 0.02 nM T07663 CPA3D1 57403394 Ki = 20800 nM T07663 CEN5Z8 57403417 IC50 = 0.08 nM T07663 CY75FP 57403418 IC50 = 0.05 nM T07663 CA4KZ8 57403419 IC50 = 1.31 nM T07663 C4XMB6 58547809 IC50 > 30000 nM T07663 CEB3G9 58547814 IC50 > 30000 nM T07663 C08QVG 58547833 IC50 > 30000 nM T07663 CFVG67 58547863 IC50 > 30000 nM T07663 CYZA38 58548077 IC50 > 30000 nM T07663 CN57ZH 67426178 IC50 > 10000 nM T07663 CO8C0Z 67453423 IC50 > 2000 nM T07663 CY8J3O 68181896 IC50 = 26000 nM T07663 CUGH78 68654838 IC50 = 1000 nM T07663 CH2X0Z 69394992 IC50 = 2.884 nM T07663 CC43LF 71074083 IC50 = 437 nM T07663 C4P0XT 71092344 IC50 = 4610 nM T07663 C6DAG4 71092519 IC50 = 13900 nM T07663 C2HGI7 71153408 IC50 > 10000 nM T07663 C9GR3L 71153436 IC50 > 10000 nM T07663 CHLQ31 71530755 IC50 = 160 nM T07663 CN8KP5 71575273 IC50 = 0.27 nM T07663 C4GNJ3 71598545 IC50 > 1000 nM T07663 C0M9IA 71666277 IC50 = 21.6 nM T07663 C3O9KX 71666278 IC50 = 0.59 nM T07663 CU0M5P 71666433 IC50 = 0.19 nM T07663 CZC74T 71666437 IC50 = 1.55 nM T07663 C68SDB 71719394 IC50 = 1995.26 nM T07663 CF2W4Z 71738037 IC50 = 240 nM T07663 C95QWN 71765666 IC50 = 17 nM T07663 CZ0G2X 72165213 IC50 > 10000 nM T07663 C7XRY6 72190879 IC50 > 30000 nM T07663 CQ3GD7 72704434 Ki = 630 nM T07663 C9JE6M 75815419 IC50 = 54.3 nM T07663 C65ZBN 76323083 IC50 = 537.03 nM T07663 CZ3P5K 89706867 IC50 = 0.056 nM T07663 CF03DW 90168772 IC50 > 20000 nM T07663 CM6J9K 90168778 IC50 > 20000 nM T07663 C45QVJ 91668196 IC50 = 2300 nM T07663 C1JPD6 91844700 IC50 = 5400 nM T07663 CYQV05 92471958 IC50 = 410 nM T07663 C6TD3W 117685212 IC50 = 337 nM T07663 CVUC27 117685328 IC50 = 1.5 nM T07663 C71BEL 117824219 IC50 = 1.7 nM T07663 CFAG87 117824250 IC50 = 0.059 nM T07663 C62NZT 117824353 IC50 = 64 nM T07663 C3WT5R 117824368 IC50 = 0.29 nM T07663 CGH1Z4 117824420 IC50 = 333 nM T07663 CX12RS 117824489 IC50 = 3.8 nM T07663 CS97IT 117830474 IC50 = 45.2 nM T07663 C60ADH 117830507 IC50 = 57 nM T07663 CMJR74 117830513 IC50 = 0.32 nM T07663 CSCY01 117949009 IC50 = 9800 nM T07663 CYQ74R 118479645 IC50 > 10000 nM T07663 CVYK24 118556943 IC50 > 50000 nM T07663 CM6XW1 118724093 IC50 = 520 nM T07663 C46LFG 118724094 IC50 > 10000 nM T07663 CYM21X 118724095 IC50 = 2900 nM T07663 C4HI1Q 118729758 IC50 = 3000 nM T07663 CKBG19 118729759 IC50 = 3100 nM T07663 C8LRQ7 121370930 IC50 = 110 nM T07663 CRJE23 122185011 IC50 > 30000 nM T07663 CS6M9C 122193679 IC50 > 100000 nM T07663 CVX7U9 127029185 IC50 = 3810 nM T07663 C9OVF8 127029366 IC50 = 5.2 nM T07663 C4UR7D 127038167 IC50 > 1000 nM T07663 C4H2TJ 127038168 IC50 > 1000 nM T07663 CL9JT8 127038169 IC50 = 606 nM T07663 CJPX60 127038509 IC50 = 232 nM T07663 C26EAG 127038511 IC50 = 201 nM T07663 CTM9E4 127038512 IC50 = 279 nM T07663 C6AQ2U 127038513 IC50 = 195 nM T07663 CV1FM0 127038868 IC50 = 228 nM T07663 CADU23 127038869 IC50 = 91.6 nM T07663 CACJ46 132489333 IC50 = 5.6 nM T07663 C2P1IU 134129996 IC50 > 100000 nM T07663 CLE03O 134130328 IC50 > 100000 nM T07663 CSN6J0 134130563 IC50 > 100000 nM T07663 C0A1CZ 134131162 IC50 > 100000 nM T07663 C23CYE 134814217 IC50 = 1.41 nM T07663 CHX5W7 134908214 IC50 = 91200 nM T07663 C1QMI8 135401477 IC50 = 26.92 nM T07663 C1BA7R 135406502 IC50 = 2 nM T07663 CIC0M9 135406542 IC50 = 3 nM T07663 CL6W5K 135406554 IC50 = 5.3 nM T07663 CL6YK2 135406621 IC50 = 1.1 nM T07663 C1LG3R 135406622 IC50 = 27 nM T07663 C9S5CV 135406637 IC50 = 1.4 nM T07663 C17YXR 135406983 IC50 = 5 nM T07663 C41TDB 135413523 IC50 = 3.5 nM T07663 C5JYM4 135415122 IC50 = 3 nM T07663 CN7LX8 135415142 IC50 = 1.5 nM T07663 CJG93Q 135415214 IC50 = 3.2 nM T07663 CQOL86 135417284 IC50 = 30 nM T07663 CG96MZ 135419216 IC50 = 2 nM T07663 COD5W1 135419220 IC50 = 2000 nM T07663 CBA1Q7 135419269 IC50 = 5 nM T07663 CP4HN6 135419318 IC50 = 7 nM T07663 CCXB28 135419329 IC50 = 2 nM T07663 CL8U1V 135419421 IC50 = 3.5 nM T07663 CN1CE4 135423930 IC50 = 2 nM T07663 C1GPZ3 135423938 IC50 = 0.2 nM T07663 C7A2NS 135427992 IC50 = 7.1 nM T07663 C6UFD4 135430871 IC50 = 10 nM T07663 C1Z3WH 135430893 IC50 = 8 nM T07663 CAJU63 135430952 IC50 = 50 nM T07663 CNP87H 135433645 IC50 = 330 nM T07663 C2DAG7 135433829 IC50 = 50 nM T07663 CHD03R 135433867 IC50 = 80 nM T07663 CJ0B6N 135438524 IC50 = 9.5 nM T07663 CJ9IE8 135438525 IC50 = 21 nM T07663 C94RVJ 135438569 IC50 = 0.7 nM T07663 C1A4MY 135439488 IC50 = 100 nM T07663 C0IE4A 135443738 IC50 = 200 nM T07663 C5U1NW 135444771 IC50 = 0.48 nM T07663 CF1U2Y 135451848 IC50 = 0.52 nM T07663 C0DBS7 135452901 IC50 = 1.905 nM T07663 CFKO84 135455980 IC50 = 5.7 nM T07663 CQW8U9 135456038 IC50 = 1 nM T07663 C9LD5N 135456042 IC50 = 2.089 nM T07663 C0BQH8 135456061 IC50 = 10 nM T07663 CA83SQ 135456100 IC50 = 1 nM T07663 C4ZQ1W 135456180 IC50 = 1.3 nM T07663 CM1K9A 135456702 IC50 = 150 nM T07663 C3R8SE 135457869 IC50 = 5200 nM T07663 C6TO5S 135462289 IC50 = 4 nM T07663 CUX8S3 135462319 IC50 = 70 nM T07663 C7HC3R 135462338 IC50 = 2.5 nM T07663 CA8X3R 135462413 IC50 = 1.7 nM T07663 CY3A0S 135462886 IC50 = 2.89 nM T07663 CA9V7D 135463722 IC50 = 10 nM T07663 C4C3JV 135467743 IC50 = 6 nM T07663 CTN73W 135467948 IC50 = 1 nM T07663 CHSI34 135469671 IC50 = 10 nM T07663 CAR9X0 135474505 IC50 = 0.62 nM T07663 CADL53 135475879 IC50 = 40 nM T07663 C3IT7F 135477808 IC50 = 13 nM T07663 C9E5KR 135480166 IC50 = 20 nM T07663 CZ9HT7 135480403 IC50 = 1.7 nM T07663 CJS37E 135482260 IC50 > 101000 nM T07663 CUNL35 135484025 IC50 = 10 nM T07663 C95GLJ 135484081 IC50 = 0.69 nM T07663 CVTR78 135484097 IC50 = 1.04 nM T07663 CKP9T0 135485820 IC50 = 5.3 nM T07663 CUV8L0 135485839 IC50 = 1.1 nM T07663 C23SWA 135485841 IC50 = 1.6 nM T07663 C4ILF7 135487662 IC50 = 1.7 nM T07663 CEHK47 135487696 IC50 = 2.6 nM T07663 CEZ5P3 135487732 IC50 = 5 nM T07663 C18DSI 135489339 IC50 = 34 nM T07663 CHO1Z5 135489408 IC50 = 7 nM T07663 CBW5A9 135491781 IC50 = 3.6 nM T07663 CG82XZ 135491934 IC50 = 18.2 nM T07663 CMNE87 135491938 IC50 = 8.2 nM T07663 CLFQ43 135493551 IC50 = 3 nM T07663 C8L1NK 135494369 IC50 = 3 nM T07663 C7FM8V 135494393 IC50 = 2 nM T07663 C3D4IY 135496441 IC50 = 3 nM T07663 C2MTZ8 135497265 IC50 = 2 nM T07663 CS4NM0 135501101 IC50 = 2 nM T07663 CJ3XM0 135503009 IC50 = 14.7 nM T07663 C86THJ 135503803 IC50 = 1 nM T07663 CN4BY1 135503843 IC50 = 2 nM T07663 C7BM8D 135504134 IC50 = 70 nM T07663 CK0S3E 135505670 IC50 = 0.9 nM T07663 C4ZNY0 135505809 IC50 = 7 nM T07663 C78CIT 135505815 IC50 = 12 nM T07663 CM27YS 135506900 IC50 = 40 nM T07663 CC87SI 135510018 IC50 = 53 nM T07663 CVM2R1 135513834 IC50 = 50 nM T07663 C6GNF4 135513951 IC50 = 0.1 nM T07663 CC9N6X 135513970 IC50 = 1 nM T07663 CL1W4B 135513981 IC50 = 5 nM T07663 CYS04P 135514690 IC50 = 0.9 nM T07663 C4NSC9 135515154 IC50 = 4 nM T07663 C9IU6B 135515212 IC50 = 2.5 nM T07663 CEV79B 135515565 IC50 = 5.5 nM T07663 C0STP6 135518654 IC50 = 2.5 nM T07663 CKDH83 135518785 IC50 = 0.2 nM T07663 C8VT4S 135520162 IC50 = 6.4 nM T07663 CKD97I 135520170 IC50 = 13 nM T07663 CL0HD1 135520500 IC50 = 18 nM T07663 C5EBI4 135525517 IC50 = 44 nM T07663 CD84SI 135528161 IC50 = 35 nM T07663 CYF17I 135528172 IC50 = 3.3 nM T07663 CB6H4I 135528567 IC50 = 13 nM T07663 C6KQV1 135528758 IC50 = 5 nM T07663 CFN34H 135528775 IC50 = 4 nM T07663 CLU8A5 135529022 IC50 = 1.53 nM T07663 C6YF2L 135529725 IC50 = 8 nM T07663 CJIA83 135529861 IC50 = 20 nM T07663 CTX70E 135530119 IC50 = 2.7 nM T07663 CCM89A 135530700 IC50 = 8.5 nM T07663 C43HNQ 135531347 IC50 = 1.1 nM T07663 CV34FU 135532825 IC50 = 5.2 nM T07663 CM3GD7 135532874 IC50 = 10 nM T07663 CGWS52 135532916 IC50 = 2.47 nM T07663 CEF96L 135536692 IC50 = 30 nM T07663 CKC9M0 135536718 IC50 = 40 nM T07663 C6E0BM 135536759 IC50 = 7 nM T07663 CWRQ95 135536783 IC50 = 4 nM T07663 C1Z7AY 135536802 IC50 = 0.8 nM T07663 CSO34W 135536977 IC50 = 0.78 nM T07663 CR0VL3 135543052 IC50 = 3.7 nM T07663 C45LHQ 135543089 IC50 = 2.76 nM T07663 CX4H6D 135544114 IC50 = 9.1 nM T07663 C4ASW0 135544141 IC50 = 0.6 nM T07663 CYE4C5 135544159 IC50 = 8 nM T07663 CW53FT 135545949 IC50 = 0.31 nM T07663 CK5F9W 135546517 IC50 = 1000 nM T07663 C9VKC6 135547908 IC50 = 10.8 nM T07663 C3HTJ7 135548164 IC50 = 3 nM T07663 C2CXY7 135559102 IC50 = 17 nM T07663 C8HW0M 135565273 IC50 = 8.9 nM T07663 C6J2FV 135566412 IC50 = 110 nM T07663 CHDC83 135566745 IC50 = 1.6 nM T07663 C5S7PD 135566746 IC50 > 1000 nM T07663 C3H1QO 135566795 IC50 = 18.2 nM T07663 CN1OH0 135566796 IC50 = 77 nM T07663 C9IJK1 135566935 IC50 = 90.6 nM T07663 C7M1TE 135604959 IC50 = 5 nM T07663 C6I3HM 135678134 IC50 = 20 nM T07663 CCB89G 135723513 IC50 = 20 nM T07663 CZP1J0 135731499 IC50 = 100 nM T07663 C7VBI4 135740146 IC50 = 82 nM T07663 CIQ83H 135744761 IC50 = 300 nM T07663 C97IUH 135750162 IC50 = 37000 nM T07663 CG1AN3 135790070 IC50 = 200 nM T07663 CD5J1S 135790088 IC50 = 1.76 nM T07663 C0M1LQ 135790105 IC50 = 0.31 nM T07663 CH13EW 135832627 IC50 = 4466.84 nM T07663 C31VFB 135832642 IC50 = 4400 nM T07663 C3PO9K 135856789 IC50 = 7560 nM T07663 C7KDO8 135874585 IC50 = 150 nM T07663 C51XVI 135874586 IC50 = 60 nM T07663 CWT6F3 135890114 IC50 = 5.8 nM T07663 C1EP3X 135890118 IC50 = 6.6 nM T07663 C25PUK 135890126 IC50 = 41 nM T07663 CI4DB0 135890131 IC50 = 4.5 nM T07663 CO07ZA 135890143 IC50 = 1.23 nM T07663 CBI80F 135890150 IC50 = 1.61 nM T07663 CQ8CT6 135890151 IC50 = 4 nM T07663 C8I2XR 135890178 IC50 = 1.01 nM T07663 CTX54Z 135896326 IC50 = 1500 nM T07663 CK4X2F 135898900 IC50 = 100 nM T07663 CPNJ62 135898901 IC50 = 50 nM T07663 C43ZKU 135898902 IC50 = 320 nM T07663 CSO02I 135898910 IC50 = 200 nM T07663 C30ZQG 135898911 IC50 = 510 nM T07663 CJQ74U 135898912 IC50 = 38 nM T07663 C4TRA9 135898925 IC50 = 70 nM T07663 CM2T5C 135898926 IC50 = 140 nM T07663 CH5R6Y 135898941 IC50 = 70 nM T07663 CYJ07O 135898942 IC50 = 530 nM T07663 CR30YL 135898943 IC50 = 500 nM T07663 C0MUP5 135898944 IC50 = 310 nM T07663 CT1H3Q 135898959 IC50 = 370 nM T07663 CU3MH0 135964375 IC50 = 381 nM T07663 CI46LV 135964379 IC50 = 1050 nM T07663 C61SDR 135964388 IC50 > 10000 nM T07663 C42FTR 135964389 IC50 = 116 nM T07663 CZ5UD9 135964390 IC50 = 710 nM T07663 CUQ41O 135964394 IC50 = 2100 nM T07663 C7NRJ6 135964396 IC50 = 849 nM T07663 CY6LT4 135964400 IC50 = 4870 nM T07663 C8UT0J 135964407 IC50 = 634 nM T07663 C04IQT 135964410 IC50 = 2160 nM T07663 C98BHJ 135964418 IC50 = 3340 nM T07663 CS4FT5 135964421 IC50 = 80 nM T07663 CO51CW 135964422 IC50 = 146 nM T07663 CC3HS1 135964423 IC50 = 15 nM T07663 C7KI6V 135964424 IC50 = 1330 nM T07663 C1WB6M 135964425 IC50 = 112 nM T07663 CKSO87 135964426 IC50 = 48 nM T07663 CY24DM 135964428 IC50 = 33 nM T07663 CMYW62 135964429 IC50 = 9 nM T07663 CPL92J 135964430 IC50 = 1570 nM T07663 CLX28E 135964433 IC50 = 38 nM T07663 C6D0FX 136026515 IC50 > 10000 nM T07663 CL7BE5 136032221 IC50 = 1.7 nM T07663 C9OQ5U 136032222 IC50 = 2.1 nM T07663 C6OU3Z 136034782 IC50 = 10 nM T07663 CWPB32 136034783 IC50 = 878 nM T07663 C3KCA0 136042216 IC50 = 0.69 nM T07663 CO4FS2 136042217 IC50 = 0.75 nM T07663 C5MCV8 136042218 IC50 = 2.44 nM T07663 C0EZ4B 136042219 IC50 = 0.74 nM T07663 CX1L3V 136042220 IC50 = 0.86 nM T07663 CS32WP 136042221 IC50 = 0.26 nM T07663 C21HJT 136042222 IC50 = 1.27 nM T07663 C4DP9X 136042223 IC50 = 1.83 nM T07663 CMH5B3 136042224 IC50 = 1.36 nM T07663 CMW86G 136042225 IC50 = 1.01 nM T07663 CJ5X4O 136042226 IC50 = 1.66 nM T07663 CM1TU5 136042227 IC50 = 4.35 nM T07663 C4A6JD 136043740 IC50 = 3.1 nM T07663 CS38OR 136044186 IC50 = 0.58 nM T07663 C6LT3U 136053630 IC50 = 0.29 nM T07663 C9OTF5 136053631 IC50 = 0.28 nM T07663 C5ZIU7 136056125 IC50 = 1000 nM T07663 C70DJG 136056126 IC50 = 2.1 nM T07663 C9Q3BW 136056127 IC50 = 81.28 nM T07663 C4U1SF 136056128 IC50 = 954.99 nM T07663 CI8E5F 136056129 IC50 = 780 nM T07663 CJ43ZC 136059652 IC50 = 3 nM T07663 CZT97J 136059653 IC50 = 77 nM T07663 C2DQ4L 136059654 IC50 = 100 nM T07663 CJ1TW7 136059659 IC50 = 80 nM T07663 CE75BO 136059660 IC50 = 100 nM T07663 C58IEH 136059684 IC50 = 1.1 nM T07663 CG6E8F 136059685 IC50 = 7.7 nM T07663 C97HLB 136059686 IC50 = 5.6 nM T07663 CZQ84P 136059687 IC50 = 0.62 nM T07663 CV6PU2 136059688 IC50 = 0.89 nM T07663 C12UMG 136059728 IC50 = 370 nM T07663 C6WH2S 136078534 IC50 = 10 nM T07663 CE51KZ 136079586 IC50 = 4 nM T07663 CRP24A 136087045 IC50 = 417 nM T07663 C7SUX4 136087050 IC50 = 141 nM T07663 C8UF7G 136087052 IC50 = 3300 nM T07663 C6U2FG 136104505 IC50 = 0.18 nM T07663 CB1GP4 136104506 IC50 = 0.28 nM T07663 CIC08H 136104509 IC50 = 0.41 nM T07663 C0LRM5 136104510 IC50 = 0.34 nM T07663 CNRF74 136104512 IC50 = 0.7 nM T07663 C5LXO8 136104513 IC50 = 0.32 nM T07663 C9UK1F 136132272 IC50 = 100 nM T07663 CBO5H3 136132273 IC50 = 50 nM T07663 CPY6I0 136132274 IC50 = 500 nM T07663 CDE2S8 136132275 IC50 = 300 nM T07663 CPL26N 136132276 IC50 = 1 nM T07663 C4ZBT6 136132277 IC50 = 300 nM T07663 CJ9QG1 136132278 IC50 = 5 nM T07663 C23BTX 136132279 IC50 = 20 nM T07663 C1BFD5 136132280 IC50 = 40 nM T07663 C21FVA 136180322 IC50 = 1.5 nM T07663 C41CAD 136180323 IC50 = 1.7 nM T07663 CC42DB 136180324 IC50 = 1.9 nM T07663 CGJX71 136180325 IC50 = 3.4 nM T07663 C0W3NC 136180326 IC50 = 3.9 nM T07663 CYC9Z6 136180327 IC50 = 12 nM T07663 C5EJ0K 136180328 IC50 = 32 nM T07663 CZ1JH2 136180329 IC50 = 14 nM T07663 C9OM5D 136180330 IC50 = 2.6 nM T07663 CMF1V6 136180331 IC50 = 1.6 nM T07663 C01TYU 136180332 IC50 = 16 nM T07663 CXT68L 136180333 IC50 = 13 nM T07663 CY0T8W 136180334 IC50 = 3.3 nM T07663 C1WHX6 136197281 IC50 = 0.83 nM T07663 CQW7T0 136197286 IC50 = 0.62 nM T07663 CPA8E7 136197297 IC50 = 1.21 nM T07663 CS8TV5 136197304 IC50 = 1.7 nM T07663 COTY62 136197323 IC50 = 8.8 nM T07663 C5HIL8 136197357 IC50 = 9.6 nM T07663 CE0F5T 136197398 IC50 = 1.46 nM T07663 CK2FL9 136197415 IC50 = 5.33 nM T07663 CS16YF 136197417 IC50 = 1.86 nM T07663 CN0G6U 136197445 IC50 = 0.92 nM T07663 C8TQ7A 136217455 IC50 = 3300 nM T07663 C4JCZ7 136219297 IC50 = 272 nM T07663 CE32YG 136219298 IC50 = 21.3 nM T07663 CXOM76 136236320 IC50 = 12.6 nM T07663 C65BFU 136236321 IC50 = 58 nM T07663 C96WPH 136236322 IC50 = 8.5 nM T07663 CY2NJ1 136236323 IC50 = 4.8 nM T07663 CUS40O 136236324 IC50 = 13.7 nM T07663 CS9Z1P 136236325 IC50 = 3 nM T07663 CRZ58U 136236326 IC50 = 4.8 nM T07663 C9PIO3 136236327 IC50 = 34.3 nM T07663 CSU3J2 136236328 IC50 = 7.2 nM T07663 C5KF0V 136236329 IC50 > 2000 nM T07663 CDNI42 136236330 IC50 = 312 nM T07663 CI0M5R 136236331 IC50 = 104 nM T07663 CF43SC 136236332 IC50 = 88 nM T07663 CMGK71 136236333 IC50 = 31.5 nM T07663 C9R6HE 136236334 IC50 = 65 nM T07663 C7ZU0K 136236335 IC50 = 71 nM T07663 C2BCV9 136236336 IC50 = 450 nM T07663 CO4S8B 136236337 IC50 > 2000 nM T07663 C6N2KA 136236338 IC50 = 12.5 nM T07663 CN69OZ 136239327 IC50 = 6.2 nM T07663 C63FEW 136239328 IC50 = 29.3 nM T07663 CQZR23 136244112 IC50 = 48 nM T07663 CO9M4H 136244113 IC50 = 10.2 nM T07663 CK6GB7 136244114 IC50 = 74 nM T07663 CF5BV2 136244123 IC50 = 25.5 nM T07663 C5VT4W 136244124 IC50 = 11.1 nM T07663 CZD04T 136244125 IC50 = 2.8 nM T07663 CUQA38 136244132 IC50 = 17.4 nM T07663 CILG36 136286746 IC50 = 3 nM T07663 C39WRP 136286747 IC50 = 3 nM T07663 C7ZX5O 136286761 IC50 = 48 nM T07663 C9SV6G 136645392 IC50 = 65 nM T07663 CANQ56 136645396 IC50 = 53 nM T07663 C9TGH1 136645397 IC50 = 14 nM T07663 C1F7JV 136645401 IC50 = 144 nM T07663 C32LNQ 136645404 IC50 = 149 nM T07663 C4W0IE 136645405 IC50 = 27 nM T07663 CMIU28 136645406 IC50 = 40 nM T07663 C3K2WL 136645410 IC50 = 79 nM T07663 CC1D0X 136645415 IC50 = 20 nM T07663 C02RIK 136645417 IC50 = 12 nM T07663 C8CT0Z 136645422 IC50 = 20 nM T07663 CAWT82 136645431 IC50 = 10 nM T07663 CBZ8Q1 136645433 IC50 = 22 nM T07663 C21EJD 136645435 IC50 = 2 nM T07663 C1KTV3 136645436 IC50 = 36 nM T07663 CK1B9W 136645438 IC50 = 1 nM T07663 C6QOP7 136645441 IC50 = 7 nM T07663 CMZ71T 136645444 IC50 = 10 nM T07663 CL47WS 136645445 IC50 = 3 nM T07663 C64BZR 136645447 IC50 = 44 nM T07663 C7X1UL 136645449 IC50 = 5 nM T07663 CI9ZO7 136645454 IC50 = 13 nM T07663 CA3I8S 136645455 IC50 = 2 nM T07663 CRN16W 136645457 IC50 = 1 nM T07663 CGQ92L 136645458 IC50 = 2 nM T07663 CO5DN2 136645462 IC50 = 2 nM T07663 CRPN39 136645466 IC50 = 11 nM T07663 CL5X3G 136645467 IC50 = 3 nM T07663 C48HNY 136959539 IC50 = 74 nM T07663 C1P8ZW 136959550 IC50 = 5 nM T07663 CKU95F 136966187 IC50 = 17 nM T07663 CFRG19 136985286 IC50 = 15 nM T07663 CE7F4O 136985287 IC50 = 10 nM T07663 CFPT21 136985288 IC50 = 0.5 nM T07663 CBH5Y0 136985291 IC50 = 24 nM T07663 CDAK28 136985292 IC50 = 0.6 nM T07663 CQ9XW7 136985295 IC50 = 122 nM T07663 C1M6NW 136985296 IC50 = 31 nM T07663 CJOA28 136985302 IC50 = 3 nM T07663 C8HG0E 137051684 IC50 = 2.02 nM T07663 CANS59 137136982 IC50 = 47 nM T07663 C5AE3Q 137283418 IC50 = 19 nM T07663 C0KM1X 137288419 IC50 = 2439 nM T07663 C5QIX1 137289788 IC50 = 17 nM T07663 C5X0YR 137289866 IC50 = 7 nM T07663 CU70ZB 137289868 IC50 = 207 nM T07663 CV6AN7 137289892 IC50 = 57 nM T07663 CB14CI 137289900 IC50 = 5 nM T07663 CLY69S 137289946 IC50 = 13 nM T07663 CC5HA4 137290225 IC50 = 121 nM T07663 C4RBC7 137290234 IC50 = 4 nM T07663 CKJ6Q4 137290238 IC50 = 46 nM T07663 CR53GQ 137290273 IC50 = 34 nM T07663 C8DYG6 137290344 IC50 = 13 nM T07663 C9G3JB 137292402 IC50 = 7 nM T07663 C6MXL3 137292504 IC50 = 57 nM T07663 CAZ49O 137300702 IC50 = 4 nM T07663 CGE0J6 137300703 IC50 = 165 nM T07663 CDU43L 137300704 IC50 = 11 nM T07663 CK0QG6 137300705 IC50 = 303 nM T07663 C91IPL 137300706 IC50 = 70 nM T07663 C5UYP8 137300707 IC50 = 5 nM T07663 CHSG63 137300708 IC50 = 23 nM T07663 CX57MR 137300709 IC50 = 39 nM T07663 C54KGS 137300710 IC50 = 10 nM T07663 CQD07Z 137300711 IC50 = 20 nM T07663 C3I1CB 137300712 IC50 = 38 nM T07663 C2N9VT 137348687 IC50 > 10000 nM T07663 C14DWB 137631637 IC50 = 157510 nM T07663 CML1E3 137631792 IC50 > 100 nM T07663 CA92EX 137632005 IC50 = 31 nM T07663 C5HM3W 137632322 IC50 = 17600 nM T07663 C0SGD8 137633727 IC50 = 77 nM T07663 CTRF70 137634642 IC50 > 100 nM T07663 CO7J5T 137635211 IC50 > 100 nM T07663 CF6EZ1 137635781 IC50 > 1000000 nM T07663 CKB51U 137637339 IC50 = 100000 nM T07663 CU17GD 137637935 IC50 = 5.4 nM T07663 C8RG2S 137638853 IC50 > 100 nM T07663 CA3BX6 137639488 IC50 > 100 nM T07663 C49UCG 137642312 IC50 > 100 nM T07663 C8R1GD 137644106 IC50 > 100 nM T07663 CSQ7P5 137644148 IC50 = 16 nM T07663 CM57EI 137646989 IC50 = 3.1 nM T07663 CPLM78 137647044 IC50 = 56 nM T07663 C18JOP 137647693 IC50 = 30 nM T07663 C4V8QP 137648482 IC50 = 50000 nM T07663 CSW42J 137651273 IC50 = 50 nM T07663 CH6EC3 137653604 IC50 > 100 nM T07663 CPK1J0 137654639 IC50 > 100 nM T07663 C93WRT 137655765 IC50 > 100 nM T07663 CDQ8B5 137657724 IC50 > 100 nM T07663 CY57JX 137658794 IC50 = 21 nM T07663 C2ITK1 137660715 IC50 > 100 nM T07663 CJA7I0 137662139 IC50 = 100000 nM T07663 C6KYD7 137700754 IC50 = 4010 nM T07663 CM3UF7 137700779 IC50 > 20000 nM T07663 CPTE92 138319693 IC50 = 0.32 nM T07663 C2QLX3 138393292 IC50 > 5000 nM T07663 CF3B2O 141492937 IC50 = 0.52 nM T07663 CEK54I 141492938 IC50 = 1.2 nM T07663 CMJW70 141492939 IC50 = 3.28 nM T07663 CKB05G 141492943 IC50 = 0.53 nM T07663 CU6A0R 141492944 IC50 = 2.85 nM T07663 CW7NV6 141492945 IC50 = 0.6 nM T07663 C2NW6Y 141492955 IC50 = 0.67 nM T07663 C13PVI 141492968 IC50 = 0.6 nM T07663 C42GOU 141492970 IC50 = 26.9 nM T07663 CGNK49 141492971 IC50 = 0.82 nM T07663 CXN3U7 141492981 IC50 = 86 nM T07663 CZ0M1Y 141492988 IC50 = 1.25 nM T07663 C2T8GE 141492992 IC50 = 6.45 nM T07663 C5XTB1 141492998 IC50 = 2.5 nM T07663 C93ZIQ 141492999 IC50 = 0.39 nM T07663 CUXZ06 141493000 IC50 = 0.97 nM T07663 C7RTX9 141493002 IC50 = 3.14 nM T07663 CQV0B4 141737648 IC50 = 155 nM T07663 C0JV6Y 141737649 IC50 = 39.7 nM T07663 CSOF52 141737655 IC50 = 19.9 nM T07663 C7SRA2 141737657 IC50 = 7.02 nM T07663 CE1H7F 141737660 IC50 = 97.5 nM T07663 CA5UL8 141737663 IC50 = 61 nM T07663 C6ZA7D 141737664 IC50 = 36.9 nM T07663 CMIY07 141737666 IC50 = 21.4 nM T07663 CC61SD 141737667 IC50 = 30.3 nM T07663 C14CZJ 141737668 IC50 = 8.44 nM T07663 CTNG49 141737674 IC50 = 36.4 nM T07663 CJ38IC 141737676 IC50 = 12.7 nM T07663 C1MC5Z 141737681 IC50 = 8.68 nM T07663 CK34HF 141737682 IC50 = 50.2 nM T07663 CQCM72 141737683 IC50 = 177 nM T07663 C2MEL1 141737684 IC50 = 56.4 nM T07663 CTUL23 141737690 IC50 = 5.24 nM T07663 CMW20N 141737696 IC50 = 3.87 nM T07663 CZWD98 141737697 IC50 = 80.2 nM T07663 C7GBH6 141737698 IC50 = 52.5 nM T07663 CVQJ85 141737699 IC50 = 383 nM T07663 CO1C4S 141737703 IC50 = 27.6 nM T07663 CX9N1P 141737704 IC50 = 10.5 nM T07663 C8HEG7 141737705 IC50 = 2.92 nM T07663 C8OWX3 145964082 IC50 = 2.64 nM T07663 C0P7CN 145964738 IC50 = 3.04 nM T07663 CZ1M5C 145964966 IC50 = 1.58 nM T07663 C07GTQ 145966108 IC50 = 0.79 nM T07663 C38QXR 145966233 IC50 = 251.19 nM T07663 CUM0Y5 145968257 IC50 = 6.82 nM T07663 CO4N2T 145968939 IC50 = 2.09 nM T07663 CDHG23 145971317 IC50 = 9.63 nM T07663 CMNV65 145973708 IC50 = 1.05 nM T07663 CC7HN2 145974174 IC50 > 100000 nM T07663 CIFW03 145974279 IC50 = 0.52 nM T07663 CWM49T 145974605 IC50 = 1.63 nM T07663 C2JF3R 145974856 IC50 = 2.64 nM T07663 C8BEH3 145975382 IC50 = 2.38 nM T07663 C5C6NR 145976885 IC50 = 2.37 nM T07663 CTJ6L8 145977069 IC50 = 0.39 nM T07663 C6M5ZW 145977440 IC50 = 19.95 nM T07663 CDB1E7 145977898 IC50 = 4.38 nM T07663 CK1BR0 145978345 IC50 > 100000 nM T07663 CJD7B2 145978603 IC50 = 4.03 nM T07663 CU5VD3 145978669 IC50 = 3.82 nM T07663 C9LGT4 145979889 IC50 = 235 nM T07663 CKZ1Y6 145979895 IC50 = 170 nM T07663 C50DFR 145982956 Ki = 8 nM T07663 CKTF58 145987769 IC50 = 227 nM T07663 CJA1B0 145991631 IC50 = 81.2 nM T07663 CHJ79V 145997874 IC50 = 3390 nM T07663 CM7TX2 148279038 IC50 = 1530 nM T07663 CYPW78 155510908 IC50 = 1.55 nM T07663 C6VZ5O 155514730 IC50 = 1.69 nM T07663 CL8CU6 155521936 IC50 > 200000 nM T07663 CAUO07 155524955 IC50 = 0.54 nM T07663 CT85RG 155530589 IC50 > 200000 nM T07663 CXMU51 155537188 IC50 = 0.79 nM T07663 C1IP4D 155556194 IC50 = 3.9 nM T07663 C2DA1W 155561694 IC50 > 500000 nM T07663 CQ2R0W 155568588 IC50 > 500000 nM T07663 CV07RN 44579973 IC50 = 0.6166 nM T07663 D00REK 5712 IC50 = 31900 nM T07663 D01RLF 105078 IC50 = 794.33 nM T07663 D01TOR 667555 IC50 = 450 nM T07663 D02NWF 2573787 IC50 = 720 nM T07663 D02VRN 6442679 IC50 = 1470 nM T07663 D03BWH 44587253 IC50 = 360 nM T07663 D06NIT 135564899 IC50 = 349 nM T07663 D06TLQ 5488822 IC50 = 1700 nM T07663 D09AUL 10266864 IC50 = 260 nM T07663 D09RKU 46239428 Ki = 9700 nM T07663 D09WUP 25058047 IC50 = 74 nM T07663 D0I6XA 149784 Ki > 200000 nM T07663 D0J0CB 2753 IC50 = 7150 nM T07663 D0J7GF 780643 IC50 = 320 nM T07663 D0O3QI 10356247 IC50 = 4200 nM T07663 D0R6MT 3758 IC50 = 63000 nM T07663 D0S8AV 509245 IC50 = 16230 nM T07663 D0U8YQ 921562 IC50 = 310 nM T07663 D0V1CL 37015 IC50 = 180 nM T07663 D0V4WB 149790 IC50 > 16000 nM T07663 D0W2BI 9799499 IC50 = 700 nM T07663 D0X7SR 10246505 IC50 = 1290 nM T07663 D0YZ0L 44605341 IC50 = 12600 nM T61657 D02DGU 444795 Ki = 0.4 nM T61657 D0BM5G 5381 EC50 = 0.8 nM T61657 D0G3PI 449171 Ki = 0.5 nM T61657 D0JC9N 60164 EC50 = 2 nM T61657 D0N0RU 82146 Ki = 50 nM T61657 D02GTY 108143 Ki = 30 nM T61657 D06FOU 11518241 EC50 = 125 nM T61657 D06QXI 9863342 EC50 = 340 nM T61657 D09YFJ 135411 EC50 = 226 nM T61657 D0M5EC 1714884 EC50 = 125.89 nM T61657 D08GRF 5287705 Ki = 0.7 nM T61657 D0YO4D 3922 Ki > 1000 nM T61657 C7QAB1 2418 EC50 = 1650 nM T61657 CZBJ59 119342 Ki = 3 nM T61657 CX90MS 128016 Ki = 680 nM T61657 CWZY65 135754 Ki = 13 nM T61657 CRJ7K2 164456 Ki = 26 nM T61657 CF61YU 2063335 EC50 = 15.85 nM T61657 CE8H3O 2757304 EC50 = 63.1 nM T61657 CLY2T6 2802556 EC50 = 100 nM T61657 CI8NO1 3025917 EC50 = 570 nM T61657 C4ZB0M 3086355 EC50 = 25.12 nM T61657 C81XYO 3092138 EC50 = 15.85 nM T61657 C0D8UF 3563820 EC50 = 31.62 nM T61657 C7AJR4 4433908 EC50 = 63.1 nM T61657 CUL8F1 5354022 EC50 = 2200 nM T61657 C8ES5G 6366138 EC50 = 190 nM T61657 C5EOB6 6366685 EC50 > 5 nM T61657 CGL71X 6366726 EC50 = 23 nM T61657 C5EON6 6366727 EC50 > 0.001 nM T61657 C62YGF 6366732 EC50 > 0.001 nM T61657 CK4UA6 6366733 EC50 = 1080 nM T61657 CLF4M5 6366734 EC50 = 21 nM T61657 CA5GS8 6438168 EC50 > 0.001 nM T61657 C7C9SR 6439768 EC50 > 10000 nM T61657 CV6S9Y 6439770 EC50 = 0.4 nM T61657 C8WU1N 6440217 EC50 = 15 nM T61657 CG1S2D 6440346 EC50 = 0.5 nM T61657 C5LH2R 6441236 EC50 = 2 nM T61657 CJHW10 6441985 EC50 = 74 nM T61657 CHA3C2 6447986 EC50 = 43 nM T61657 C3F4GD 6447987 EC50 = 72 nM T61657 CEV62Y 6450532 EC50 = 40 nM T61657 C31YCL 9797765 Ki = 36 nM T61657 CBE62R 9799320 EC50 > 1000 nM T61657 CRK31P 9799442 EC50 = 436 nM T61657 COP9S7 9799477 EC50 = 220 nM T61657 CENQ29 9799532 IC50 = 22 nM T61657 CSNI93 9799841 EC50 > 10000 nM T61657 CX2HY4 9801929 EC50 > 10000 nM T61657 CCUE13 9802971 Ki = 4064 nM T61657 CW7D0R 9810431 EC50 = 2068 nM T61657 CUJ14W 9819890 EC50 > 10000 nM T61657 CEK1O4 9820039 EC50 = 46 nM T61657 CQI49S 9820393 EC50 > 10000 nM T61657 C7R9JM 9820462 Ki = 90 nM T61657 C2X3PS 9822318 EC50 = 8.6 nM T61657 C9SQ7J 9825106 Ki > 10000 nM T61657 CIWO37 9843061 EC50 = 25 nM T61657 CI1P9A 9844563 Ki = 156 nM T61657 CQFA96 9845057 Ki = 4687 nM T61657 CE7D1J 9845382 IC50 = 6.5 nM T61657 CQ1ZH6 9847065 Ki = 2270 nM T61657 C4W3MR 9864378 EC50 = 200 nM T61657 CA74MZ 9864886 IC50 = 40 nM T61657 C2ZY0W 9865875 EC50 > 1000 nM T61657 CZVA73 9866726 Ki > 10000 nM T61657 C8F3DE 9867254 Ki > 10000 nM T61657 CAE0R3 9868664 Ki = 6008 nM T61657 CRC51S 9869157 Ki = 5325 nM T61657 CA0TS6 9884959 EC50 = 139 nM T61657 CSK5B8 9885521 EC50 > 1000 nM T61657 CH0PV4 9885573 IC50 = 1000000 nM T61657 C3CS9R 9886082 EC50 > 10000 nM T61657 C5AD1H 9886137 Ki > 10000 nM T61657 C41JUL 9887430 EC50 = 115 nM T61657 CG3JR4 9887949 EC50 > 10000 nM T61657 CRA64P 9888023 Ki > 10000 nM T61657 CU2OI0 9888037 Ki = 8269 nM T61657 C8V1ON 9888385 IC50 = 7.5 nM T61657 C90UXQ 9889347 Ki = 5681 nM T61657 C8MK1Y 9889522 Ki = 320 nM T61657 C2WFX1 9905729 EC50 = 304 nM T61657 C2D9WJ 9906413 EC50 = 2238 nM T61657 C9AJZ7 9906514 EC50 = 17 nM T61657 C7E0IO 9907433 EC50 > 10000 nM T61657 CK9Z7I 9907650 IC50 = 230 nM T61657 CVG53F 9910801 Ki = 8000 nM T61657 C0A3UZ 9911319 Ki = 2112 nM T61657 CSW2Y8 9929026 EC50 = 339 nM T61657 C9WZ1S 9930650 Ki = 5623 nM T61657 CTXK14 9932151 Ki > 10000 nM T61657 CX7U3M 9932436 Ki = 8064 nM T61657 CIS1Z0 9948900 EC50 = 355 nM T61657 C9VEF0 9949645 EC50 = 1388 nM T61657 C6CI3S 9950957 EC50 > 10000 nM T61657 CS8M7V 9953061 EC50 = 26 nM T61657 CU46RB 9953712 Ki = 71 nM T61657 C6JLI1 9973307 EC50 > 10000 nM T61657 CV1A3K 9974457 EC50 > 1000 nM T61657 C63OUJ 9976842 EC50 > 1000 nM T61657 CT7YJ8 9977495 EC50 > 1000 nM T61657 C05EXS 9998870 EC50 > 10000 nM T61657 CL7X4Y 9999621 EC50 > 10000 nM T61657 CM1BQ5 10003577 Ki = 3927 nM T61657 CZP71W 10022432 EC50 = 310 nM T61657 CN6LP5 10022568 EC50 > 10000 nM T61657 C4K5OP 10026035 Ki = 4742 nM T61657 C6L0XH 10044201 Ki = 36 nM T61657 CN0Y1P 10044591 EC50 = 45 nM T61657 CC4MF5 10045395 EC50 = 92 nM T61657 CE60FI 10065757 EC50 = 287 nM T61657 C2C0GJ 10066739 EC50 = 29 nM T61657 CVMD62 10069273 EC50 = 41 nM T61657 C4VU6T 10087372 EC50 > 10000 nM T61657 CC8R9M 10093918 Ki = 320 nM T61657 C8MG7C 10094345 IC50 > 3000 nM T61657 CSG68Q 10127015 IC50 = 22 nM T61657 C72HLB 10172878 IC50 = 21 nM T61657 C15HAE 10194688 IC50 = 15 nM T61657 C9XS2G 10203771 Ki = 288 nM T61657 CVL1Q6 10227224 Ki = 89 nM T61657 C3IHN5 10251128 IC50 = 25 nM T61657 CSE96Y 10292425 IC50 = 250000 nM T61657 CY1J5M 10308975 Ki > 1000 nM T61657 C9D7QC 10314719 EC50 = 0.3 nM T61657 C7G6XH 10315687 EC50 = 3 nM T61657 CVQ7Z6 10316839 EC50 > 10000 nM T61657 C6C5GP 10320109 Ki = 810 nM T61657 C5LV9X 10358286 EC50 = 1200 nM T61657 CUEF37 10362997 IC50 = 150 nM T61657 CG01ED 10383375 EC50 = 337 nM T61657 CIK6T7 10384337 EC50 = 256 nM T61657 CW39AL 10384413 IC50 = 53 nM T61657 CJCA73 10385620 Ki = 1245 nM T61657 C25HLM 10389354 Ki = 158 nM T61657 CTO46Q 10405813 IC50 = 140 nM T61657 CXQ9S4 10450790 EC50 = 395 nM T61657 CXA0N9 10458226 Ki = 500 nM T61657 CV7C4F 10478196 IC50 = 2 nM T61657 C0KZT7 10519016 Ki = 105 nM T61657 CY62NU 10523459 Ki = 70 nM T61657 CQR8K0 10524574 IC50 = 4.5 nM T61657 C5BXE0 10543210 EC50 > 1000 nM T61657 CUO1I2 10543981 Ki = 12 nM T61657 C6CWZ1 10545954 EC50 = 110 nM T61657 C26NJB 10547547 IC50 = 2.5 nM T61657 C9EBZ0 10572606 IC50 = 36 nM T61657 CKBI92 10619546 IC50 = 39 nM T61657 CS96IV 10619935 EC50 = 31 nM T61657 C2HXP8 10641611 Ki = 90 nM T61657 CMH87P 10643692 EC50 > 10000 nM T61657 CZ2C5K 10663499 Ki > 3000 nM T61657 C92TJP 10666483 Ki = 17 nM T61657 CSC54U 10687664 EC50 > 1000 nM T61657 C89VQU 10690943 IC50 = 290 nM T61657 C9K4YM 10709275 EC50 > 1000 nM T61657 C1SNV6 10760998 Ki = 660 nM T61657 C9UFH8 10763649 Ki = 105 nM T61657 C2TJY4 10788561 Ki > 10000 nM T61657 CTI5N7 10789247 Ki = 21 nM T61657 CMXI39 10804037 EC50 = 770 nM T61657 C4U5ZQ 10906425 Ki = 2056 nM T61657 C8UG3F 10926235 EC50 > 500 nM T61657 C13TFH 10938920 Ki > 10000 nM T61657 C75PWJ 10961406 Ki > 10000 nM T61657 CL9QM1 11070809 Ki > 10000 nM T61657 CV38KY 11167904 EC50 = 13 nM T61657 CW14SH 11253452 EC50 > 100000 nM T61657 C27ERO 11279584 IC50 = 90000 nM T61657 CX24ON 11317250 EC50 = 7700 nM T61657 CT4HL6 11340230 IC50 = 32000 nM T61657 CZ8IT7 11349121 IC50 = 175000 nM T61657 CUY07B 11382535 IC50 = 500000 nM T61657 CCL2D4 11472545 EC50 > 100000 nM T61657 CY6PJ9 11504066 EC50 = 40 nM T61657 CJH04T 11510627 EC50 = 35 nM T61657 CM34CL 11518525 EC50 = 14 nM T61657 C9NH8Y 11547131 EC50 = 25 nM T61657 CQAF21 11554936 EC50 = 17 nM T61657 CLID54 11569584 EC50 = 9.5 nM T61657 CQ8S3K 11627002 EC50 = 60 nM T61657 C41AJB 11634244 EC50 > 10000 nM T61657 C3RMA0 11718697 EC50 = 248 nM T61657 C34NCO 11724776 EC50 > 1000 nM T61657 C0S9KJ 11740691 EC50 = 1004 nM T61657 CFC0X5 11751490 IC50 < 1 nM T61657 C7H2KQ 11784536 EC50 = 17600 nM T61657 C0WA5F 11793407 EC50 = 8 nM T61657 CD5K4U 11799011 Ki > 10000 nM T61657 C7UWV3 12112296 EC50 = 21 nM T61657 CIQJ20 12112298 EC50 = 21 nM T61657 CQ9YE5 12358678 EC50 = 3.3 nM T61657 C97MLN 13554588 EC50 = 50.12 nM T61657 CL23YP 13765519 EC50 = 1000 nM T61657 C7JSH9 13833722 EC50 = 140 nM T61657 C1M8SC 13833726 EC50 = 430 nM T61657 C7Z0YT 13833727 EC50 = 320 nM T61657 CT41DZ 14557465 EC50 = 1900 nM T61657 CN7CX1 14726558 IC50 = 100 nM T61657 C8DP6M 14776682 EC50 = 18 nM T61657 CQI17S 15160092 EC50 = 5 nM T61657 CNS9T8 15434197 Ki > 1000 nM T61657 CS2B4X 15951828 EC50 = 100 nM T61657 CU8LV5 15951923 EC50 = 39.81 nM T61657 CDA7J9 15951925 EC50 = 63.1 nM T61657 C4LRI8 15951927 EC50 = 63.1 nM T61657 C9S5XT 15952013 EC50 = 79.43 nM T61657 CCZ8Y4 15952016 EC50 = 125.89 nM T61657 CKW7N6 15952017 EC50 = 125.89 nM T61657 C0AZ9Q 15952019 EC50 = 100 nM T61657 CX2CS8 15952020 EC50 = 251.19 nM T61657 C3U7WJ 15952211 EC50 = 630.96 nM T61657 C5J3ZE 16661643 EC50 = 6.8 nM T61657 CX6L0G 16661644 EC50 = 3.8 nM T61657 C5GTA2 18507967 EC50 = 250 nM T61657 CQYD01 18768139 EC50 = 5 nM T61657 CX3Q7D 20243100 EC50 = 0.4 nM T61657 C5MHX3 21217837 Ki > 3000 nM T61657 CV1C4A 22226112 EC50 > 1000 nM T61657 CLV67T 22971725 EC50 = 10 nM T61657 CTE1N2 24748569 EC50 > 10000 nM T61657 C26ZLQ 25259039 EC50 < 10000 nM T61657 C1TH9L 25259040 EC50 < 10000 nM T61657 CSTR97 25259041 EC50 = 39.81 nM T61657 CP6OG5 25259262 EC50 < 10000 nM T61657 C7FLT0 25259263 EC50 < 10000 nM T61657 CT2B1Z 25259265 EC50 = 19.95 nM T61657 C2G6QF 25259266 EC50 = 56.7 nM T61657 C4HJ5Z 25259267 EC50 < 10000 nM T61657 CO7M0D 44285104 EC50 = 1100 nM T61657 CS7U6L 44285287 EC50 = 20 nM T61657 CFTB98 44313143 Ki > 3000 nM T61657 C4E1OW 44313513 Ki > 3000 nM T61657 C8W6JP 44314319 Ki = 11 nM T61657 C17LMT 44314320 Ki > 1100 nM T61657 C7U3IB 44316094 EC50 = 1000 nM T61657 CRY69X 44316095 EC50 = 36 nM T61657 COX51B 44316155 EC50 = 280 nM T61657 C92VTZ 44316277 EC50 = 170 nM T61657 C8RM3G 44316292 EC50 = 4 nM T61657 C90NSH 44316354 EC50 = 4 nM T61657 CIVH74 44316525 Ki > 1000 nM T61657 CAP68W 44316543 EC50 = 809 nM T61657 CAI2Z5 44316544 Ki > 1000 nM T61657 C0YQ8H 44316756 Ki > 1000 nM T61657 C6Q1CA 44316796 EC50 = 637 nM T61657 CLK5H0 44316811 EC50 = 559 nM T61657 CK48CT 44321880 EC50 = 3200 nM T61657 CID72B 44321881 EC50 = 2000 nM T61657 CXV0B4 44321951 EC50 = 1500 nM T61657 C1KUN0 44325759 Ki > 1000 nM T61657 CLB6X7 44325767 EC50 = 809 nM T61657 CW0T6K 44353336 Ki = 2112 nM T61657 C8K0AB 44353347 Ki = 4623 nM T61657 C3DYE9 44353422 Ki = 3597 nM T61657 C5DTY3 44353441 Ki = 1956 nM T61657 C2M8TN 44353456 Ki > 10000 nM T61657 CVKA40 44353466 Ki = 2612 nM T61657 C8J5SA 44353480 Ki = 1984 nM T61657 CIB15X 44353481 Ki > 10000 nM T61657 C3MY4C 44364348 Ki = 210 nM T61657 CY9XP2 44366042 EC50 > 10000 nM T61657 CT3S5O 44377822 EC50 = 8 nM T61657 COX1B7 44397758 EC50 = 5300 nM T61657 C5QRI4 44401302 IC50 = 7 nM T61657 CJVG73 44459626 EC50 = 1800 nM T61657 CR5SI0 44476535 EC50 > 10000 nM T61657 CP4DM5 44581289 EC50 = 10 nM T61657 C8UHG5 45270032 IC50 = 40 nM T61657 CUD91T 49862248 EC50 > 10000 nM T61657 C5ZX4B 54597874 EC50 > 10000 nM T61657 C9G4IT 60729785 EC50 = 77.8 nM T61657 CZ38NM 69588033 EC50 = 40 nM T61657 CN03UB 71568951 EC50 = 136.3 nM T61657 CX9EA0 71568952 EC50 = 12.1 nM T61657 C4GRK9 71571262 EC50 = 11 nM T61657 C6TBD2 121345502 EC50 > 20000 nM T61657 CQZ9W3 121414283 EC50 = 2.05 nM T61657 C6L4GM 135949402 EC50 = 26 nM T61657 C5L6AU 136126668 EC50 = 820 nM T61657 CN5MO3 136126669 EC50 > 1000 nM T61657 CJ5EH7 136126670 EC50 > 1000 nM T61657 CI4CG1 136126671 EC50 > 1000 nM T61657 C1J4DV 145965542 EC50 = 2.5 nM T61657 CRKW68 145966900 EC50 > 10000 nM T61657 C4MY5N 145967331 EC50 = 26 nM T61657 CC05VW 145970742 EC50 > 10000 nM T61657 CDBR75 145976745 EC50 = 40 nM T61657 C2A1UC 10429766 Ki > 1000 nM T61657 D09RRF 11530459 EC50 = 7.943 nM T61657 D0F8CC 10090192 EC50 = 140 nM T61657 D0F8JO 9951075 IC50 = 175000 nM T61657 D0G6JM 5289501 Ki = 0.5 nM T61657 D0P0PP 10044792 IC50 = 135 nM T61657 D0Q0IR 177238 IC50 = 20 nM T61657 D0Q9FZ 6442223 EC50 = 10 nM T61657 D0RD0R 2126 EC50 = 8.6 nM T61657 D0X5WP 10410894 Ki = 220 nM T37541 D00STL 644241 Ki = 99 nM T37541 D01MUR 68844 Ki = 2.8 nM T37541 D01WLC 4170 Ki = 2.1 nM T37541 D02PJA 24841 Ki = 250000 nM T37541 D03QGM 5355 Ki = 3.6 nM T37541 D03RTS 2662 Ki = 2170 nM T37541 D03UOT 785 Ki = 883000 nM T37541 D04AIT 5280445 Ki = 4.7 nM T37541 D05OFX 219078 Ki = 4446 nM T37541 D05UYW 5284549 Ki = 3.5 nM T37541 D07HBX 338 Ki = 82100 nM T37541 D07INV 3295 Ki = 0.78 nM T37541 D07MGA 72281 Ki = 3.3 nM T37541 D07VDZ 5284627 Ki = 0.87 nM T37541 D09NIA 2732 Ki = 2.8 nM T37541 D09VAZ 5565 Ki = 45000 nM T37541 D0AZ3C 5291 Ki = 109 nM T37541 D0AZ8C 5213 Ki = 4710 nM T37541 D0C2II 4100 Ki = 2.1 nM T37541 D0C8FX 3005837 Ki = 7760 nM T37541 D0E1SW 1986 Ki = 2 nM T37541 D0H8FH 3702 Ki = 0.23 nM T37541 D0J4GO 3038 Ki = 6 nM T37541 D0J7RK 36811 Ki = 4300 nM T37541 D0K0OZ 5702160 Ki = 3 nM T37541 D0K1QD 3998 Ki = 75 nM T37541 D0K8KX 5280343 Ki = 4840 nM T37541 D0L4JT 5333 Ki = 70 nM T37541 D0L6DA 119607 Ki = 3900 nM T37541 D0OT0O 44561 Ki = 560000 nM T37541 D0PQ3G 3440 Ki = 513 nM T37541 D0SH3I 387447 Ki = 6940 nM T37541 D0U5QK 1983 Ki = 9100 nM T37541 D0W5HK 216239 Ki = 8136.4 nM T37541 D0Y2IZ 5560 Ki = 7.9 nM T37541 D0Z3EI 6038 Ki = 420 nM T37541 D04IIU 216468 Ki = 122 nM T37541 D04PBH 5280804 Ki = 3.8 nM T37541 D05NJI 5287541 Ki = 23 nM T37541 D08BXT 1102 Ki = 1230 nM T37541 D0I7MT 5281807 Ki = 452.6 nM T37541 D0L6HN 996 Ki > 500000 nM T37541 D0U3EP 445154 Ki = 4350 nM T37541 D0V0UK 82267 Ki = 6800 nM T37541 D03SLR 445858 Ki = 7410 nM T37541 D0NH9P 135 Ki = 4080 nM T37541 D0X2AU 23427 Ki > 100000 nM T37541 D0LD9S 1103 Ki = 710 nM T37541 CI0WH9 72 Ki = 7870 nM T37541 CUT2V4 260 Ki = 1060000 nM T37541 COV5W3 402 Ki = 1240000 nM T37541 CSZ43B 540 Ki = 15200000 nM T37541 C97QXH 767 Ki = 160000 nM T37541 C39CTO 768 Ki = 9200000 nM T37541 C1QDT0 781 Ki = 170000 nM T37541 CW0R2L 944 Ki = 190000 nM T37541 CQV86E 1100 Ki = 7300000 nM T37541 C8W7BZ 1118 Ki = 1380000 nM T37541 CU12QE 1203 Ki = 450 nM T37541 C6O0MZ 1491 Ki = 72000 nM T37541 C5L7VX 2871 Ki = 4680 nM T37541 CQ0D8J 3469 Ki = 68000 nM T37541 CJ2F6P 5056 Ki = 8980 nM T37541 CDJ4K6 5987 Ki = 9500 nM T37541 CUP2F4 7043 Ki = 7250 nM T37541 C1CVT7 7121 Ki = 7150 nM T37541 C6NC4O 7414 Ki = 5740 nM T37541 C6QYD8 8434 Ki = 8700 nM T37541 CHP7I1 9016 Ki = 3880 nM T37541 CLYZ50 9338 Ki = 6600 nM T37541 CV5PC3 11568 Ki = 5900 nM T37541 CUA0L6 14917 Ki = 1240000 nM T37541 CNI85U 15109 Ki = 3220 nM T37541 CQ4C5U 16523 Ki = 850 nM T37541 CNGB21 20098 Ki = 900 nM T37541 C3LA1Z 20161 Ki = 940 nM T37541 C3NG2U 24529 Ki = 1780000 nM T37541 CFM9L6 24530 Ki = 1410000 nM T37541 C3F1OY 25502 Ki = 670000 nM T37541 C4OU6D 35703 Ki = 7800 nM T37541 CN94KU 65008 Ki = 8870 nM T37541 C1NQ8E 65188 Ki = 9180 nM T37541 CT6YO0 66548 Ki = 6270 nM T37541 C0ZK7U 67284 Ki = 3700 nM T37541 CVI38F 69809 Ki = 410 nM T37541 CTMF08 75076 Ki = 780 nM T37541 C0I4UT 75077 Ki = 8300 nM T37541 CE5RZ1 76509 Ki = 730 nM T37541 C9V0ME 77547 Ki = 750 nM T37541 C6TS8J 77548 Ki = 830 nM T37541 CX79KD 78297 Ki = 273.1 nM T37541 CX47BZ 78479 Ki = 58000 nM T37541 C5BFK4 87432 Ki = 700 nM T37541 C6K3MG 101424 Ki > 100000 nM T37541 CN19UT 129695 Ki = 100 nM T37541 C2P0RH 139584 Ki = 36540000 nM T37541 CJ0FR9 155148 Ki = 9310 nM T37541 C8AO0Z 165323 Ki = 5.4 nM T37541 CU3WG6 179620 Ki = 8850 nM T37541 CSMP84 219987 Ki = 470 nM T37541 C3QV5H 287064 Ki = 810 nM T37541 C26HNY 289493 Ki = 9030 nM T37541 C96DKW 310360 Ki = 8550 nM T37541 CT3ZU4 388776 Ki = 1090 nM T37541 CH21KA 389641 Ki = 107000 nM T37541 C6CQO3 389642 Ki = 108000 nM T37541 CNPZ40 394897 Ki = 35 nM T37541 C7HME8 439246 Ki = 4.3 nM T37541 CA8C5N 439514 Ki = 9110 nM T37541 C5HM8E 474578 Ki = 465.8 nM T37541 C49CNT 519869 Ki = 710 nM T37541 CJ7FR6 533728 Ki = 1470000 nM T37541 CYGK68 676946 Ki = 850 nM T37541 CMO61A 694792 Ki = 7.1 nM T37541 CF93TC 821388 Ki = 810 nM T37541 C8SN5L 889524 Ki = 51 nM T37541 CEN67I 897592 Ki = 861 nM T37541 C4QX1Z 1146666 Ki = 2.6 nM T37541 C6T0NU 1230924 Ki = 9.5 nM T37541 C9IBF8 1241259 Ki = 0.74 nM T37541 CF1N3S 1277269 Ki = 4 nM T37541 C40CKN 1316238 Ki = 3.2 nM T37541 C9DY2L 1488548 Ki = 380 nM T37541 CDQR23 2049187 Ki = 9.8 nM T37541 C2O9YS 2196398 Ki = 6.5 nM T37541 C4TD8M 2388085 Ki = 1.3 nM T37541 C8QGL9 2760606 Ki > 10000 nM T37541 CE2GR3 2900806 Ki = 1240 nM T37541 CME74N 2904589 Ki = 605 nM T37541 C61OTP 2991092 Ki = 21 nM T37541 CN2Y5M 3083616 Ki = 5560 nM T37541 C9GT5Z 3083928 Ki = 9280 nM T37541 CL6E2Y 3426384 Ki = 5122 nM T37541 CQ5F9P 3724005 Ki = 9.5 nM T37541 CV0KG3 3950536 Ki = 4.3 nM T37541 C4E5VQ 4447263 Ki = 5.8 nM T37541 C96LCZ 4476238 Ki = 65 nM T37541 CDK4L0 4608376 Ki = 600000 nM T37541 CLSY09 4626049 Ki = 760 nM T37541 C3GDR0 4634582 Ki = 62 nM T37541 CCB9Z5 4656684 Ki = 71 nM T37541 C7JBU0 5019114 Ki = 161 nM T37541 C4OAL9 5070078 Ki = 6400 nM T37541 CI8JY0 5172475 Ki = 4.3 nM T37541 CY9IV8 5223338 Ki = 5 nM T37541 CEBD92 5272990 Ki = 4600 nM T37541 CP09FG 5272997 Ki = 5900 nM T37541 C4SV5T 5273568 Ki = 3870 nM T37541 CU4E5S 5273569 Ki = 4320 nM T37541 CN10FM 5281793 Ki = 71.4 nM T37541 CA18OQ 5316302 Ki = 4530 nM T37541 CTJ01E 5317485 Ki = 8110 nM T37541 CI58XK 5319562 Ki = 820 nM T37541 CNO53D 5321265 Ki = 650 nM T37541 C8PS4E 5358858 Ki = 3690 nM T37541 CXEW32 5491996 Ki = 14500 nM T37541 CK0M4A 5910585 Ki = 7820 nM T37541 C2JTF7 6432768 Ki = 5010 nM T37541 CS4KQ6 6482974 Ki = 7010 nM T37541 C9L8AX 6537802 Ki = 840 nM T37541 C65FRB 6852128 Ki = 6.4 nM T37541 CKCM96 7463376 Ki = 7950 nM T37541 CDCP43 7766335 Ki = 630 nM T37541 CY47OI 9998322 Ki = 6.5 nM T37541 CNKD31 10016330 Ki = 620.3 nM T37541 C5X7GY 10059582 Ki = 1899 nM T37541 CY8F0E 10076040 Ki = 58300 nM T37541 C0P5XV 10081897 Ki = 956 nM T37541 CD58EL 10083644 Ki = 720 nM T37541 C7WU0A 10107532 Ki = 467.8 nM T37541 CJV68L 10220266 Ki = 389.3 nM T37541 CQ8A0I 10328097 Ki = 26.6 nM T37541 CN40WD 10331524 Ki = 1178 nM T37541 C3HBY6 10375558 Ki = 66 nM T37541 CVIN94 10439991 Ki = 4.7 nM T37541 CWQY26 10535227 Ki > 10000 nM T37541 C73KXU 10586607 Ki = 14500 nM T37541 C9TSQ6 10632698 Ki = 31400 nM T37541 C6D2TJ 10712038 Ki = 35 nM T37541 C36BAC 11034581 Ki > 100000 nM T37541 C8C6ER 11069133 Ki = 2.9 nM T37541 CMK4Y0 11096006 Ki = 435.5 nM T37541 CIL4M9 11183499 Ki > 100000 nM T37541 CHC42Y 11245700 Ki = 19 nM T37541 CF15AS 11287957 Ki = 4965 nM T37541 CHA0V5 11321514 Ki = 910 nM T37541 C8PM3Z 11353795 Ki = 18 nM T37541 CM8P2L 11609292 Ki = 23 nM T37541 C9QL2F 11615432 Ki = 7507 nM T37541 C9JR2I 11674590 Ki = 8580 nM T37541 CV7HN1 11795548 Ki = 15 nM T37541 CNHD71 12051191 Ki > 200000 nM T37541 CMPA32 12066940 Ki > 500000 nM T37541 CB15KR 12066941 Ki > 500000 nM T37541 C60EFT 12354987 Ki = 300 nM T37541 C5RS4H 12528487 Ki = 975.3 nM T37541 CM8TP6 12528490 Ki = 1364 nM T37541 CK90BP 12765315 Ki = 320 nM T37541 CF2BM7 13177311 Ki = 2.1 nM T37541 C8VM1A 13201770 Ki = 720 nM T37541 CC25BI 13927398 Ki = 1100000 nM T37541 C7K4JV 14024589 Ki = 1282 nM T37541 C4UG2O 14057643 Ki > 100000 nM T37541 CHOG93 14611919 Ki = 89 nM T37541 C76ASY 14787919 Ki > 200000 nM T37541 CH5YR2 15014351 Ki > 200000 nM T37541 C7XD2T 15118768 Ki = 8980 nM T37541 CK8GE9 15230629 Ki = 1790 nM T37541 C8PMQ9 15729847 Ki > 200000 nM T37541 C8PER5 15938557 Ki > 500000 nM T37541 C3W2MB 15939939 Ki = 3.9 nM T37541 CC0Z4V 16119626 Ki = 730 nM T37541 CDWU20 17537594 Ki = 39.4 nM T37541 CK7D2I 17748220 Ki = 10 nM T37541 CLY1N4 17757567 Ki = 170 nM T37541 C6SFI8 18268734 Ki = 4.7 nM T37541 CR9VF3 18668331 Ki = 9.9 nM T37541 CQE5K4 18710120 Ki > 200000 nM T37541 C60NAV 18971452 Ki = 86.4 nM T37541 C2K5BX 19374444 Ki = 8.3 nM T37541 C62PKT 19838794 Ki = 7.8 nM T37541 CDU40W 20184392 Ki > 200000 nM T37541 CKR8T2 20970546 Ki = 10.5 nM T37541 C61KUX 21726402 Ki = 1.7 nM T37541 CJ4O2E 21806575 Ki = 5.8 nM T37541 C02IPY 21978067 Ki = 10.1 nM T37541 C9U4TE 22313850 Ki = 135 nM T37541 C9KMP4 23275795 Ki = 7.7 nM T37541 C7V6YP 23665706 Ki = 0.24 nM T37541 C01LHS 24640776 Ki = 13.3 nM T37541 CT8O2Z 24643222 Ki = 9.5 nM T37541 CISH83 25186263 Ki = 1.5 nM T37541 CU14KG 25258358 Ki = 68700 nM T37541 CQ1WE2 25258360 Ki > 200000 nM T37541 CL5EZ6 25258361 Ki > 200000 nM T37541 COU19V 25258363 Ki > 200000 nM T37541 CRP6F5 25335375 Ki = 62.9 nM T37541 CPN2T5 25392418 Ki = 6.9 nM T37541 C5EC2T 26535209 Ki = 10.4 nM T37541 CLNR46 26598995 Ki = 3238 nM T37541 CA9UZ7 26773685 Ki = 6.9 nM T37541 CI0K1J 36865965 Ki = 8.3 nM T37541 C6WU8M 42609905 Ki = 2.7 nM T37541 CYJ0H4 43089860 Ki = 16.5 nM T37541 CIM4Z8 43132043 Ki = 5.4 nM T37541 CXJY80 43235186 Ki = 4.6 nM T37541 C7EO2A 43329592 Ki = 8.9 nM T37541 CA0DX4 43342474 Ki = 9.7 nM T37541 C2HY4R 43342475 Ki = 9.4 nM T37541 CBK0M6 43342481 Ki = 0.9 nM T37541 C82MRL 44144383 Ki = 73.2 nM T37541 CI3O9B 44395149 Ki = 45 nM T37541 CMSJ40 44395790 Ki = 3.7 nM T37541 CZ4DF9 44399462 Ki = 8.3 nM T37541 CD5MJ6 44399571 Ki = 9.4 nM T37541 C2T7MB 44399654 Ki = 84 nM T37541 CA90GQ 44424362 Ki = 160 nM T37541 C5HB4P 44424363 Ki > 200000 nM T37541 CK8S7Y 44424364 Ki > 200000 nM T37541 C28QYE 44424366 Ki = 320 nM T37541 CM3J0U 44430517 Ki = 24 nM T37541 C9LT7Y 44430518 Ki = 41 nM T37541 C1VTB6 44430520 Ki = 79 nM T37541 C2L5MB 44430521 Ki = 18 nM T37541 CVEO17 44430523 Ki = 23 nM T37541 C8MFL1 44430524 Ki = 25 nM T37541 CFW8V2 44520897 Ki = 7 nM T37541 CR4NZ3 44520898 Ki = 6.9 nM T37541 CI78UO 44520899 Ki = 7.2 nM T37541 CQUC34 44520900 Ki = 6.9 nM T37541 CNC1D8 44520905 Ki = 8.5 nM T37541 CR43NP 44520906 Ki = 6.1 nM T37541 CXD9V3 44590306 Ki > 200000 nM T37541 COE8U0 45267045 Ki = 35.5 nM T37541 C23MVW 45269009 IC50 = 27900 nM T37541 C0RG8K 45269749 Ki = 8500 nM T37541 CSW5V6 45378228 Ki = 6.4 nM T37541 CV5RQ3 45484187 Ki = 98 nM T37541 CTG20B 45485271 Ki = 8900 nM T37541 CK4U0V 45485283 Ki = 3200 nM T37541 C6ION5 46236927 Ki = 49 nM T37541 C7SFG3 46236928 Ki = 8370 nM T37541 CC82QE 46237039 Ki = 556 nM T37541 CBCK34 46237040 Ki = 60 nM T37541 CSD29O 46237041 Ki = 581 nM T37541 CEB1X9 46237042 Ki = 54 nM T37541 C1VIK9 46237043 Ki = 53 nM T37541 C3RJ5M 46237044 Ki = 5150 nM T37541 CU5Y9E 46237045 Ki = 6.5 nM T37541 CM7N6J 46237172 Ki = 64 nM T37541 CP15GJ 46237173 Ki = 54 nM T37541 CT65RE 46868356 Ki = 3.9 nM T37541 CNEO10 46871889 Ki = 4.6 nM T37541 C93AIR 46899573 Ki = 108000 nM T37541 CJ0R2O 46911381 Ki = 48 nM T37541 C0NUM6 53386724 Ki = 60.2 nM T37541 C54FGU 53386866 Ki = 12.1 nM T37541 CRI54V 53386867 Ki = 34.9 nM T37541 CUX7S4 53386868 Ki = 91.7 nM T37541 CCFP92 53516400 IC50 > 50000 nM T37541 C6SM5T 54613427 Ki = 7 nM T37541 C0ZJ2L 55629711 Ki = 310 nM T37541 CIJ9V0 56684131 Ki = 912 nM T37541 CH52DA 56921864 Ki = 6750 nM T37541 CTFL92 56928044 Ki = 10.2 nM T37541 C4VGE9 57047254 Ki = 8.3 nM T37541 CP7YR5 57345662 Ki = 270 nM T37541 C1M0LS 57394809 Ki = 690 nM T37541 CW1TU4 57412422 Ki = 4.8 nM T37541 CT4BV9 57412423 Ki = 5.9 nM T37541 C31NWX 57412424 Ki = 13.9 nM T37541 CD86ER 57412425 Ki = 6.5 nM T37541 CB94YU 57412426 Ki = 8 nM T37541 C2K8YJ 57412507 Ki = 5.7 nM T37541 CSF4V6 57412508 Ki = 5.8 nM T37541 CHAO86 57412509 Ki = 8.2 nM T37541 C3U6TH 57412510 Ki = 34.7 nM T37541 C40LOS 57412511 Ki = 23.4 nM T37541 CZ47VT 57412512 Ki = 17.8 nM T37541 C28WRD 57412600 Ki = 61.7 nM T37541 C2XPG5 57413583 Ki = 7.9 nM T37541 CM2AY7 57413584 Ki = 50.8 nM T37541 C9V6EY 60446869 Ki = 911.3 nM T37541 CGF3W6 66586679 Ki = 890 nM T37541 CN84CU 66586879 Ki = 840 nM T37541 C2Y5KV 70682044 Ki = 73.3 nM T37541 CXJ16H 71450117 Ki = 873 nM T37541 CB8JA3 71455488 Ki = 628 nM T37541 C02UHX 71455489 Ki = 609 nM T37541 CICJ97 71457274 Ki = 602 nM T37541 CMHG14 71521493 Ki = 6300 nM T37541 CHN53G 71521494 Ki = 7100 nM T37541 CZJ5M6 71521495 Ki = 5800 nM T37541 CFBE53 71521496 Ki = 4900 nM T37541 CME27W 71521497 Ki = 9000 nM T37541 C24XWU 71521575 Ki = 9500 nM T37541 CJF68W 71521576 Ki = 9300 nM T37541 C19OIY 71579130 Ki = 730 nM T37541 CGO24R 71584196 Ki = 465 nM T37541 CV0LU6 71602117 Ki = 540 nM T37541 CZL96Y 71602476 Ki = 3.1 nM T37541 C50LSJ 71714068 Ki = 24900 nM T37541 CM4T1R 71717003 Ki = 78400 nM T37541 CG4I1X 71718239 Ki = 7200 nM T37541 C0LYX1 71718858 Ki = 4300 nM T37541 CM24ND 71719433 Ki = 800 nM T37541 CT3D5S 71719441 Ki = 6800 nM T37541 CJG34A 71720036 Ki = 6920 nM T37541 CIU4L2 71720670 Ki = 8700 nM T37541 C0ROQ1 71770179 Ki = 3.5 nM T37541 C8W6DJ 71770180 Ki = 3.5 nM T37541 CB3Y0X 71770181 Ki = 46.9 nM T37541 CKHM42 71770182 Ki = 1.3 nM T37541 CBL41T 71770183 Ki = 4.7 nM T37541 C30EYH 71770184 Ki = 2.2 nM T37541 C5IU0Y 72163201 Ki = 54 nM T37541 CNP42E 72163326 Ki = 4 nM T37541 C2KE5D 72163327 Ki = 55 nM T37541 C0Q5XL 72163343 Ki = 59 nM T37541 C63MIX 72163344 Ki = 77 nM T37541 CL3WV2 72163345 Ki = 80 nM T37541 C4T9DA 72163346 Ki = 175 nM T37541 CTK07O 72163347 Ki = 84 nM T37541 CE32BF 72163348 Ki = 72 nM T37541 CBN48K 72163465 Ki = 65 nM T37541 CGB02D 72163466 Ki = 199 nM T37541 CVFN85 72163467 Ki = 41 nM T37541 C82RDA 72163468 Ki = 245 nM T37541 CA1X6Z 72163476 Ki = 68 nM T37541 C7TKJ4 72163610 Ki = 368 nM T37541 C70OBD 72163611 Ki = 264 nM T37541 CA0Q4T 72163612 Ki = 152 nM T37541 C96GMR 72163613 Ki = 127 nM T37541 CJ2K8R 72163743 Ki = 498 nM T37541 CPY81U 72163744 Ki = 334 nM T37541 CC1D3Y 72163745 Ki = 225 nM T37541 CYH0G5 72163746 Ki = 375 nM T37541 CEZM40 72163861 Ki = 5 nM T37541 CMBR85 72163862 Ki = 14 nM T37541 CZ9IE5 72163863 Ki = 22 nM T37541 CZM75P 72163975 Ki = 142 nM T37541 CPT0C9 72163976 Ki = 46 nM T37541 CX82JD 72696463 Ki = 6.2 nM T37541 COCV73 72696591 Ki = 21.9 nM T37541 C5KHD7 72696592 Ki = 8.5 nM T37541 C4FBA6 72696593 Ki = 6.7 nM T37541 CO1JM5 72696594 Ki = 6.5 nM T37541 CUF61Q 72696595 Ki = 8.3 nM T37541 CO1JT3 73054728 Ki = 30 nM T37541 CU9I6V 82078731 Ki = 125.5 nM T37541 C5TB6O 82080973 Ki = 690.9 nM T37541 C6UZR9 82911195 Ki = 9.6 nM T37541 C3AYZ5 91811067 Ki = 2796 nM T37541 CQF98O 91827503 Ki = 8.5 nM T37541 C3I6NV 91827505 Ki = 9.2 nM T37541 CW1P4E 91827506 Ki = 819 nM T37541 C28QRZ 101564149 Ki > 100000 nM T37541 CDGZ03 101879106 Ki = 24 nM T37541 CY6ER7 101879108 Ki = 17.7 nM T37541 CB1PK8 102151146 Ki > 100000 nM T37541 C0A6FY 102151151 Ki = 7800 nM T37541 C1XV9H 102311866 Ki = 8900 nM T37541 C0CVO4 102480165 Ki > 100000 nM T37541 CUR4V8 114816322 Ki = 0.27 nM T37541 CKV43U 118710106 Ki = 303.5 nM T37541 CBAQ59 118710108 Ki = 269 nM T37541 C0D1SQ 118724328 Ki = 50.6 nM T37541 C89YTC 118724329 Ki = 253.5 nM T37541 CBT87C 118724330 Ki = 28.7 nM T37541 C49AWZ 118724331 Ki = 21.9 nM T37541 CHE1K4 118729473 Ki = 8.9 nM T37541 C9V8MA 118729474 Ki = 97.2 nM T37541 C8GJP5 118729475 Ki = 70.7 nM T37541 C4MEZ0 118729476 Ki = 73.8 nM T37541 CE3IV5 118729477 Ki = 8.6 nM T37541 CUQ7H9 119082247 Ki = 40.5 nM T37541 CN16RY 122189300 Ki = 2.4 nM T37541 CYN3T8 122189301 Ki = 878 nM T37541 CSW9D1 122189302 Ki = 3.1 nM T37541 C6USQ7 122189303 Ki = 2.8 nM T37541 CQ4X1G 122189304 Ki = 4 nM T37541 CH1N0C 122193189 Ki = 730 nM T37541 C19HVL 122193190 Ki = 820 nM T37541 C5TQJ1 122193251 Ki = 520 nM T37541 C8XCL0 122193252 Ki = 710 nM T37541 CC1UO6 122226187 Ki = 660 nM T37541 C7T0FH 122226188 Ki = 1800 nM T37541 C3EG2B 122226189 Ki = 6500 nM T37541 C26IUP 122386532 Ki > 100000 nM T37541 CV4GW7 126961712 Ki = 0.21 nM T37541 C0FD4E 126961713 Ki = 0.19 nM T37541 CS2K4U 127034999 Ki = 0.24 nM T37541 CFG39M 127035855 Ki = 0.43 nM T37541 C6MH2V 127035856 Ki = 0.45 nM T37541 CVO4B6 127035857 Ki = 2.2 nM T37541 CQC6P9 127035858 Ki = 0.31 nM T37541 C7YA3N 127035859 Ki = 0.3 nM T37541 CXZI89 127035860 Ki = 0.28 nM T37541 C5KLP8 127035861 Ki = 0.37 nM T37541 CL76JS 127037630 Ki = 0.39 nM T37541 CY1JU3 127037755 Ki = 5.1 nM T37541 C0UQ7W 127037756 Ki = 3.3 nM T37541 CQUE67 127037757 Ki = 3.5 nM T37541 CG8B3V 127039153 Ki = 0.46 nM T37541 CIO74C 127039154 Ki = 0.35 nM T37541 C0L8NH 127039155 Ki = 0.31 nM T37541 CS96GU 127039479 Ki = 4.4 nM T37541 C3J8ET 127040041 Ki = 2.9 nM T37541 CQC6A4 127042329 Ki = 14.5 nM T37541 C5EX6R 127048632 Ki = 48.2 nM T37541 CK1X5H 127048994 Ki = 2 nM T37541 C2XK0I 127048995 Ki = 1.3 nM T37541 CY4P2X 127048996 Ki = 5.7 nM T37541 C6JB5S 127048997 Ki = 90.7 nM T37541 C1T3WG 127049310 Ki = 39 nM T37541 CKO03S 127049970 Ki = 44.6 nM T37541 CP8KG9 127049971 Ki = 10.4 nM T37541 C9EJ6L 127050230 Ki = 22.4 nM T37541 C7MI5Q 127050568 Ki = 29.6 nM T37541 C1RGQ6 127050569 Ki = 28.9 nM T37541 CB5W0L 127050570 Ki = 10.9 nM T37541 CUG58A 127050571 Ki = 35 nM T37541 C9FZ4E 127050900 Ki = 8.1 nM T37541 CUWE95 127051804 Ki = 50.5 nM T37541 COBU26 127051805 Ki = 60.7 nM T37541 C7SIY6 127051806 Ki = 50 nM T37541 CJ7WT3 127052106 Ki = 35.5 nM T37541 C26TUM 127052712 Ki = 8.5 nM T37541 C7PS8D 127052713 Ki = 54.8 nM T37541 C32ART 127052714 Ki = 54.6 nM T37541 C9D6CB 127053004 Ki = 22.6 nM T37541 CHN5K6 127567366 Ki = 198.5 nM T37541 C4JC3W 127573780 Ki = 801.2 nM T37541 CXN16P 132495328 Ki = 0.8 nM T37541 CKLY32 132502995 Ki = 1881.2 nM T37541 C5O1JE 132547793 Ki > 100000 nM T37541 CKYC42 132547798 Ki > 100000 nM T37541 CRL24F 132596304 Ki > 50000 nM T37541 C4K1YW 132961363 Ki = 6.7 nM T37541 CQ64ZM 132961364 Ki = 3.8 nM T37541 C5LGV6 132961365 Ki = 4.5 nM T37541 C69NDK 133107891 Ki = 0.27 nM T37541 C2AIR8 134129901 Ki = 0.81 nM T37541 C1Y9AL 134130029 Ki = 0.68 nM T37541 CU10DE 134130177 Ki = 9.1 nM T37541 CP8XK0 134130364 Ki = 4 nM T37541 C83LZE 134130471 Ki = 1.8 nM T37541 C5N8AO 134130483 Ki = 7.2 nM T37541 C9V3LX 134130512 Ki = 6.4 nM T37541 CO7G6J 134130566 Ki = 0.91 nM T37541 C69IZA 134130639 Ki > 10000 nM T37541 C8MGN3 134130817 Ki = 65.3 nM T37541 C52IRH 134131086 Ki = 0.7 nM T37541 C9HVL2 134131189 Ki = 0.73 nM T37541 C7GBW5 134131361 Ki = 9.1 nM T37541 C3WJR8 134131535 Ki = 3.6 nM T37541 CQ0K5P 134131567 Ki = 1.4 nM T37541 C8Q5JZ 134131574 Ki = 7.6 nM T37541 CZQ3T2 134132041 Ki > 10000 nM T37541 C89TVU 134132755 Ki = 9.6 nM T37541 CFQG76 134133776 Ki = 8 nM T37541 CT8Z2Q 134133785 Ki = 7.4 nM T37541 CHR23F 134137004 Ki > 10000 nM T37541 C2X1UG 134137145 Ki = 51.9 nM T37541 CHM19B 134139215 Ki = 26.8 nM T37541 CRNF42 134140829 Ki = 62 nM T37541 C1T9JU 134140936 Ki = 52.2 nM T37541 CG4NU1 134141378 Ki = 5.7 nM T37541 CIK25S 134142323 Ki = 67.1 nM T37541 CIRG86 134142877 Ki = 7.8 nM T37541 CWT6O9 134142989 Ki = 29 nM T37541 C5BD1C 134143174 Ki > 10000 nM T37541 CWQ62J 134144541 Ki = 1000 nM T37541 CG7X9K 134144756 Ki = 49.1 nM T37541 CJ5QD3 134144926 Ki = 602.5 nM T37541 CR5F8T 134145685 Ki = 423.5 nM T37541 C8FV5Y 134147016 Ki > 10000 nM T37541 C0TV9S 134147261 Ki = 308.3 nM T37541 C85ABV 134147911 Ki = 54.6 nM T37541 CGBZ05 134148709 Ki = 4.1 nM T37541 CS7K8C 134149271 Ki = 701.1 nM T37541 CD5TI1 134149815 Ki = 628.7 nM T37541 CZ2C3J 134149835 Ki = 3.8 nM T37541 CIL4H9 134151823 Ki > 10000 nM T37541 C9GF7L 134152087 Ki = 7 nM T37541 CZ4WI8 134152920 Ki = 86.3 nM T37541 CD4EN0 134153199 Ki = 45.3 nM T37541 CH6OT4 134153506 Ki = 27.4 nM T37541 CZ9T6I 134153525 Ki > 10000 nM T37541 CWSI54 134154346 Ki = 376.2 nM T37541 CQZU97 134154945 Ki > 10000 nM T37541 C52UTP 134156470 Ki = 4.3 nM T37541 C7OV6T 134156655 Ki = 88.9 nM T37541 CR3Q5U 134159783 Ki = 2 nM T37541 CV9W6N 134159784 Ki = 0.24 nM T37541 CJT9W0 135393499 Ki = 0.45 nM T37541 CK8FP3 135393500 Ki = 2.6 nM T37541 CRL4V7 135393501 Ki = 7.8 nM T37541 CPW4T3 135530880 Ki = 28 nM T37541 C4KH2F 136138702 Ki = 53.6 nM T37541 CYKW91 136728963 Ki = 665.3 nM T37541 CRK6Y9 137631731 Ki = 2614 nM T37541 CZ5GQ4 137631746 Ki > 100 nM T37541 CFQ5W2 137631798 Ki = 490 nM T37541 CBJ75C 137632178 Ki = 536.5 nM T37541 CYD0E3 137632442 Ki = 6.8 nM T37541 CL5K3D 137632743 Ki > 100 nM T37541 C9YKD5 137633039 Ki = 27.8 nM T37541 C5J3AX 137633409 Ki = 121.4 nM T37541 C9AD2H 137633797 Ki = 188 nM T37541 C7N0ER 137634525 Ki > 100000 nM T37541 CP0EC3 137635051 Ki = 281.6 nM T37541 CY1HI4 137635059 Ki = 892.1 nM T37541 C1ZKU2 137635320 Ki = 15.2 nM T37541 CV12YX 137636350 Ki > 100 nM T37541 C7YKB0 137636981 Ki > 50000 nM T37541 C2Z7GO 137637071 Ki = 3.8 nM T37541 C0H2CK 137637173 Ki = 10.1 nM T37541 CWO5Z6 137637365 Ki > 100 nM T37541 CGV9M8 137637508 Ki = 8683 nM T37541 CG0N8K 137637564 Ki = 408.1 nM T37541 C80KCO 137637736 Ki = 79.3 nM T37541 C2HY8G 137637767 Ki = 64.5 nM T37541 CHQ3P9 137638456 Ki = 28.6 nM T37541 CK6OW4 137638637 Ki = 0.77 nM T37541 C6V8ED 137638882 Ki = 5.4 nM T37541 C64JQN 137639095 Ki = 0.53 nM T37541 C4LB2X 137639339 Ki = 100.4 nM T37541 C0IQ1U 137639377 Ki = 4200 nM T37541 COE61G 137639833 Ki = 5800 nM T37541 C2OT9R 137640310 Ki > 50000 nM T37541 CX3JI9 137640517 Ki = 55.2 nM T37541 C6B0CQ 137641198 Ki = 0.51 nM T37541 C0HER8 137641290 Ki > 50000 nM T37541 CMOZ57 137641425 Ki = 203 nM T37541 C53ZAF 137641717 Ki > 10000 nM T37541 CR5JZ8 137642047 Ki > 10000 nM T37541 CCSN50 137642054 Ki > 100 nM T37541 CN6WS9 137642180 Ki = 8.9 nM T37541 CEOC90 137642331 Ki = 9388 nM T37541 CSY67B 137642513 Ki = 3198 nM T37541 C61TSP 137642864 Ki > 100000 nM T37541 C3Y2GU 137643607 Ki = 9.4 nM T37541 C1BW5I 137643671 Ki > 100000 nM T37541 C0B8QA 137643949 Ki > 100 nM T37541 CF31BQ 137644307 Ki = 13.2 nM T37541 CFA3R0 137644914 Ki = 605 nM T37541 C6UAB5 137645654 Ki = 5001 nM T37541 CDZ6T8 137645734 Ki = 267.6 nM T37541 CBRK83 137645944 Ki = 9.3 nM T37541 C7E6NL 137646223 Ki = 299 nM T37541 C10YVU 137646329 Ki > 50000 nM T37541 C5WG2P 137646543 Ki = 16.2 nM T37541 C0YFX2 137646956 Ki > 10000 nM T37541 CRP78K 137647221 Ki > 100 nM T37541 CXD9A0 137647636 Ki = 0.4 nM T37541 CR2H7M 137647845 Ki > 50000 nM T37541 CCD71U 137648259 Ki = 1907.3 nM T37541 C49PLO 137648279 Ki = 694.3 nM T37541 CW8CL7 137648379 Ki = 55.5 nM T37541 CK14XO 137648525 Ki = 3343 nM T37541 C21TVD 137648644 Ki = 707.1 nM T37541 C6RIM2 137648717 Ki = 67.2 nM T37541 CEZT03 137649001 Ki = 8.5 nM T37541 CI9LS2 137649321 Ki = 43.6 nM T37541 CSWR71 137649376 Ki = 911.9 nM T37541 C4N1MP 137650156 Ki = 84.4 nM T37541 CD08YK 137650293 Ki = 138.4 nM T37541 CKJ36G 137650647 Ki = 1897.6 nM T37541 CD7S5L 137650698 Ki > 100000 nM T37541 CV89IF 137651491 Ki = 90.9 nM T37541 CSTP12 137651755 Ki = 0.35 nM T37541 C01BXO 137651769 Ki > 100 nM T37541 CY0C6Z 137652226 Ki > 100 nM T37541 C6GWB1 137652305 Ki > 100 nM T37541 CN3RQ8 137652373 Ki > 10000 nM T37541 C9UGN4 137653309 Ki = 58.5 nM T37541 C8Y7XR 137653485 Ki = 85.6 nM T37541 CIV3E9 137653528 Ki = 1.7 nM T37541 CTP0U2 137654343 Ki = 91 nM T37541 CXC7I2 137655261 Ki = 88.6 nM T37541 C2P5FH 137655445 Ki = 404 nM T37541 C3DT7S 137655450 Ki > 100 nM T37541 CASB61 137655528 Ki > 100 nM T37541 CAZ27T 137655913 Ki = 54.7 nM T37541 C27ALW 137655946 Ki = 3.2 nM T37541 CC0OY9 137655984 Ki = 177.6 nM T37541 C8TJN9 137656061 Ki = 553.5 nM T37541 COEY05 137656447 Ki = 16.7 nM T37541 C0CK7G 137656796 Ki > 10000 nM T37541 C8RNZ6 137657759 Ki > 100 nM T37541 C0KI6G 137657917 Ki = 583.3 nM T37541 C41MLN 137658275 Ki > 10000 nM T37541 CKX78V 137658314 Ki = 1885.2 nM T37541 CL2H0T 137658375 Ki > 100 nM T37541 CT98MV 137658877 Ki > 100 nM T37541 C8YV5D 137659052 Ki = 0.33 nM T37541 CXO9Y7 137659205 Ki > 100 nM T37541 CJ5O8M 137659269 Ki = 360 nM T37541 C5AM2K 137659383 Ki > 10000 nM T37541 C60DEN 137660288 Ki > 10000 nM T37541 CMS92X 137660799 Ki = 1.8 nM T37541 C0TZD5 137661006 Ki > 100000 nM T37541 C0PIE6 137661027 Ki = 78.1 nM T37541 CQ56MJ 137661167 Ki = 347.5 nM T37541 C62QWK 137661307 Ki = 5065 nM T37541 CRC92Y 137661359 Ki = 0.77 nM T37541 C1Z8KG 137661675 Ki = 0.2 nM T37541 C74YSR 137661914 Ki = 37.8 nM T37541 CEAR56 137662187 Ki = 318 nM T37541 CMP8S7 137662201 Ki = 9.2 nM T37541 CFR73V 137662256 Ki = 84.5 nM T37541 CIX41M 138393379 Ki = 0.8 nM T37541 CBOM51 138753317 Ki = 0.8 nM T37541 CB83JY 139593608 Ki = 5.7 nM T37541 C8BZI0 145949366 Ki = 0.84 nM T37541 CHVR98 145949393 Ki = 74.2 nM T37541 C7X0DZ 145949728 Ki = 462.8 nM T37541 C20RXT 145949974 Ki = 1.9 nM T37541 C9QUL0 145951028 Ki = 36.2 nM T37541 CPD05I 145951366 Ki = 0.38 nM T37541 C86DBE 145951463 Ki = 6.8 nM T37541 C38QHU 145951654 Ki = 0.93 nM T37541 CIM8X0 145951670 Ki = 7.4 nM T37541 CJ2W6V 145951720 Ki = 0.25 nM T37541 C2OTU3 145951886 Ki = 3.8 nM T37541 C4N3QL 145952239 Ki = 0.77 nM T37541 CM30EN 145952365 Ki = 311.8 nM T37541 C75RDX 145952490 Ki = 4.6 nM T37541 C26OLK 145952634 Ki = 37.4 nM T37541 CW42HX 145952649 Ki = 0.97 nM T37541 C56QVF 145952880 Ki = 0.85 nM T37541 CAS8M7 145952940 Ki = 0.83 nM T37541 C5DJY9 145953324 Ki = 3.5 nM T37541 CVNE29 145954045 Ki = 86 nM T37541 CD52IH 145954185 Ki = 0.96 nM T37541 C0XO6A 145954770 Ki = 17.4 nM T37541 C1LFA9 145954917 Ki = 3.4 nM T37541 C0UG3K 145955383 Ki = 0.87 nM T37541 C89HDL 145956309 Ki = 7.2 nM T37541 CYJ3N0 145956346 Ki = 0.31 nM T37541 C2KV9S 145956347 Ki = 9.4 nM T37541 CWPZ94 145956803 Ki = 0.93 nM T37541 C7K2DA 145957040 Ki = 0.97 nM T37541 CAMD59 145957136 Ki = 7.1 nM T37541 CM07ZF 145958200 Ki = 6.6 nM T37541 CXVC18 145959110 Ki = 0.84 nM T37541 CU8J0M 145959118 Ki = 645 nM T37541 CWNS89 145959524 Ki = 0.77 nM T37541 CPL41Z 145959905 Ki = 0.71 nM T37541 CGZ1K8 145959957 Ki = 0.35 nM T37541 C2SI5J 145960220 Ki = 1.8 nM T37541 C6JND4 145960287 Ki = 0.68 nM T37541 C6JG2V 145961631 Ki = 0.28 nM T37541 CD9I1U 145971467 Ki = 27.1 nM T37541 CGE23X 145972719 Ki = 295.6 nM T37541 CSPH69 145979414 Ki = 11.4 nM T37541 CQDB02 145979430 Ki = 49.6 nM T37541 CUDO01 145979473 Ki = 135.3 nM T37541 CIF72X 145979737 Ki = 125.9 nM T37541 CLFJ74 145980146 Ki = 6.2 nM T37541 C9S0WG 145983404 Ki = 132.2 nM T37541 CB5G4W 145983664 Ki = 750.9 nM T37541 C8C0AB 145984626 Ki = 118.2 nM T37541 CN56XE 145986933 Ki = 147.7 nM T37541 CZPA17 145987454 Ki = 78.8 nM T37541 CJ1P5W 145988462 Ki = 127.4 nM T37541 C1LV0U 145988936 Ki = 606.7 nM T37541 C9RVK0 145989853 Ki = 17.8 nM T37541 CHMR39 145990191 Ki = 41.5 nM T37541 CYOD69 145990290 Ki = 98.4 nM T37541 CZB2X3 145990392 Ki = 121.5 nM T37541 CB63XC 145990519 Ki = 180.8 nM T37541 C3QXL4 145991981 Ki = 94.7 nM T37541 C7RYJ4 145992796 Ki = 147.1 nM T37541 CE34YK 145992956 Ki = 72 nM T37541 C48CZD 146160385 Ki = 16.1 nM T37541 C6FD2N 147348395 Ki = 2565 nM T37541 C1PG9M 155511036 Ki = 2.7 nM T37541 CN6DW9 155511075 Ki = 25 nM T37541 CJA94W 155512108 Ki = 0.72 nM T37541 CZ5W1M 155514230 Ki = 3589.4 nM T37541 CM5J3L 155514471 Ki = 18.1 nM T37541 CDM78Q 155514660 Ki = 18.9 nM T37541 CCQB03 155515285 Ki = 37.2 nM T37541 CT2ZB0 155515980 Ki = 1 nM T37541 CZN16J 155516304 Ki = 69 nM T37541 COP4Q6 155516517 Ki = 5.4 nM T37541 C2E0ZF 155517026 Ki = 56.4 nM T37541 CAG9L4 155517430 Ki = 3.6 nM T37541 C1VNX3 155518220 Ki = 31.4 nM T37541 CEH62Y 155518447 Ki = 5.6 nM T37541 CP7UI1 155518510 Ki = 6.2 nM T37541 C8MYG2 155519248 Ki = 12.2 nM T37541 CO6D1Y 155519288 Ki = 41.5 nM T37541 CC47MV 155519432 Ki = 85.4 nM T37541 CO4V0B 155519627 Ki = 44.4 nM T37541 CIV68R 155520019 Ki = 38.2 nM T37541 CP49HE 155520274 Ki = 4.7 nM T37541 C8E0SN 155520671 Ki = 4900 nM T37541 C4LPA1 155520806 Ki = 792.4 nM T37541 CQ0OR1 155520930 Ki > 10000 nM T37541 C2J1YG 155521041 Ki = 15.4 nM T37541 CCGT71 155521462 Ki = 3.1 nM T37541 CF7HE1 155521700 Ki = 5.8 nM T37541 CZ7WI8 155521830 Ki = 23.5 nM T37541 C6AWP0 155522679 Ki = 4.8 nM T37541 C3HGK6 155523328 Ki = 5.5 nM T37541 CSC58M 155524279 Ki > 10000 nM T37541 C9PV5X 155524649 Ki > 100000 nM T37541 CS21YC 155524712 Ki = 86.3 nM T37541 C70ZPH 155524915 Ki = 5.3 nM T37541 CA02GS 155526086 Ki = 85.5 nM T37541 CWGS97 155526825 Ki = 609 nM T37541 CAMY18 155527145 Ki = 4.3 nM T37541 CDE96Y 155527673 Ki = 55.2 nM T37541 CLF2V0 155528496 Ki = 28.6 nM T37541 C38SKR 155528605 Ki = 68.1 nM T37541 CB08MU 155528753 Ki > 100000 nM T37541 C2LF1H 155528761 Ki = 69.3 nM T37541 CN27OU 155528858 Ki = 488.1 nM T37541 CECZ45 155529036 Ki = 363.3 nM T37541 C8DN2F 155529373 Ki = 304.1 nM T37541 CG3J0Q 155529984 Ki = 55 nM T37541 CKO2V5 155530358 Ki = 71.3 nM T37541 CIGQ50 155530440 Ki = 30.4 nM T37541 CTJ3I7 155530506 Ki = 4.7 nM T37541 CO7P5W 155531268 Ki = 0.68 nM T37541 CLMZ93 155531382 Ki = 9.3 nM T37541 CW6TC5 155531936 Ki = 3100 nM T37541 C5H8QF 155532861 Ki = 893 nM T37541 C0BNY7 155533528 Ki = 52.2 nM T37541 C78ZFI 155534074 Ki = 11.9 nM T37541 CT5NG1 155534179 Ki = 0.2 nM T37541 CS0FK9 155534753 Ki = 78.7 nM T37541 CE1I8S 155535343 Ki = 273 nM T37541 CVU5P6 155535355 Ki = 1.5 nM T37541 CV0N9I 155535382 Ki > 10000 nM T37541 CKR07J 155535598 Ki > 10000 nM T37541 CNFR72 155535756 Ki > 100000 nM T37541 CFYA23 155535780 Ki = 33.9 nM T37541 CD2O3A 155535852 Ki = 810 nM T37541 CZPY79 155536184 Ki = 210.1 nM T37541 C0EDQ2 155536876 Ki = 65.1 nM T37541 CZ0T6A 155537018 Ki = 3949 nM T37541 COP2R4 155537042 Ki = 48.3 nM T37541 C4K0MB 155537772 Ki = 870 nM T37541 CYM0A3 155538069 Ki = 70.2 nM T37541 C5RV9W 155538073 Ki = 81.7 nM T37541 COX74J 155538083 Ki = 62.8 nM T37541 C9AP8F 155538224 Ki = 20.8 nM T37541 C9K2TL 155539730 Ki = 1690 nM T37541 CS1G5V 155539783 Ki = 75.5 nM T37541 CS1UR7 155539868 Ki = 78.8 nM T37541 CSAD81 155540401 Ki = 13.5 nM T37541 CZ8FJ3 155540422 Ki = 58 nM T37541 C8RV6T 155541805 Ki = 3.7 nM T37541 CW96ES 155541807 Ki = 1.1 nM T37541 C4MW9Q 155541811 Ki = 79.2 nM T37541 CZ2CT0 155542259 Ki = 534 nM T37541 CW61DF 155542555 Ki = 46.6 nM T37541 CT9GZ2 155542660 Ki = 1034.1 nM T37541 CDK2W5 155542691 Ki = 34.6 nM T37541 C75TVG 155542954 Ki = 261.9 nM T37541 C2AEH6 155543096 Ki = 355 nM T37541 CN2SJ7 155543228 Ki = 48.1 nM T37541 C19DJA 155543271 Ki = 647 nM T37541 CI2T8N 155544664 Ki = 49.4 nM T37541 CY6SX5 155545800 Ki > 100000 nM T37541 C83ZIS 155547526 Ki = 36 nM T37541 CW19PC 155547551 Ki = 94.5 nM T37541 C73YLV 155547628 Ki = 0.8 nM T37541 C61MSB 155547730 Ki = 0.78 nM T37541 CQG5F9 155548326 Ki = 15.7 nM T37541 CU1NE7 155549031 Ki = 3 nM T37541 CA25QH 155549266 Ki = 43.3 nM T37541 CR79SY 155549354 Ki = 705 nM T37541 C4O6TN 155550616 Ki = 17 nM T37541 CMWQ79 155550618 Ki = 916.3 nM T37541 C6XPV0 155550626 Ki = 85.4 nM T37541 C4S0JZ 155551334 Ki = 100.8 nM T37541 COC4Z9 155551784 Ki = 18.9 nM T37541 CZ0T3C 155551786 Ki = 3.5 nM T37541 CG9PN8 155552113 Ki = 3 nM T37541 CW8S7L 155552594 Ki = 96.4 nM T37541 C0OG8P 155553361 Ki = 0.38 nM T37541 CP15VC 155553400 Ki > 50000 nM T37541 C1R7CJ 155553759 Ki = 34 nM T37541 CMEP40 155554179 Ki = 30.5 nM T37541 CZU9Y7 155554800 Ki = 46.3 nM T37541 C5YA7C 155555084 Ki = 46.8 nM T37541 CWB82E 155555878 Ki = 5.1 nM T37541 CD4K6H 155556521 Ki = 0.55 nM T37541 CJF9O7 155557300 Ki > 100000 nM T37541 C40MOH 155557452 Ki = 2.9 nM T37541 CH1Z2S 155558695 Ki = 910 nM T37541 CXE2R9 155561928 Ki = 63.7 nM T37541 C6KD7C 155563215 Ki = 761.5 nM T37541 CP85AZ 155563623 Ki = 41.3 nM T37541 C07GFY 155564664 Ki = 80.6 nM T37541 C0E4QV 155565149 Ki = 6.1 nM T37541 CNL8B7 155565372 Ki = 584.9 nM T37541 CJ7I6Z 155565419 Ki = 7.7 nM T37541 COA9F8 155566222 Ki = 8700 nM T37541 CCW3L7 155566305 Ki = 735 nM T37541 CJQP47 155566378 Ki = 9.5 nM T37541 CI8U3W 155566755 Ki = 174.5 nM T37541 CDB8T4 155568445 Ki = 4.4 nM T37541 C94QKZ 155568447 Ki = 3323 nM T37541 CH5VU6 155568899 Ki = 4.4 nM T37541 C1C2GI 155569076 Ki = 0.63 nM T37541 C83MGT 155569151 Ki = 46.3 nM T37541 C1A7IN 155569676 Ki = 4.4 nM T37541 D00FGB 11414131 Ki = 10 nM T37541 D00GVA 44520904 Ki = 7.9 nM T37541 D00IUB 13019 Ki = 777000 nM T37541 D00RNZ 910172 Ki = 15300 nM T37541 D00XIB 11680415 Ki = 1.7 nM T37541 D00XJA 711717 Ki = 50500 nM T37541 D00YEF 148885 Ki = 92.3 nM T37541 D01BUB 94952 Ki = 554000 nM T37541 D01ISX 670786 Ki = 7.6 nM T37541 D01STY 9861037 Ki = 150 nM T37541 D01UYI 5281607 Ki = 171.41 nM T37541 D02DBP 5054 Ki = 644000 nM T37541 D02QGI 273 Ki = 420 nM T37541 D03DAM 2725651 Ki = 7200 nM T37541 D03NBX 637308 Ki = 620 nM T37541 D03ZMQ 323 Ki = 3300 nM T37541 D04CVC 4687472 Ki = 75 nM T37541 D04HRS 404195 Ki = 46 nM T37541 D04NSN 169682 Ki = 80 nM T37541 D05QOR 5280460 Ki = 8710 nM T37541 D05QUG 45485279 Ki = 44500 nM T37541 D05TLB 11117301 Ki = 76.6 nM T37541 D05WQF 637540 Ki > 1000000 nM T37541 D05XZM 10081162 Ki = 60 nM T37541 D06ALC 6441498 Ki = 268.3 nM T37541 D06DYP 234562 Ki = 32400 nM T37541 D06XNT 4119643 Ki = 6.8 nM T37541 D07CYN 20347846 Ki = 1.6 nM T37541 D07LYW 11537386 Ki = 9.3 nM T37541 D07MTM 403 Ki = 1359000 nM T37541 D07PNA 11660633 Ki = 1.9 nM T37541 D07QJJ 289 Ki = 714000 nM T37541 D07TAJ 914298 Ki = 9700 nM T37541 D07YDN 5281654 Ki = 4.4 nM T37541 D08AIJ 440735 Ki = 4.3 nM T37541 D08AOA 11543564 Ki = 3.9 nM T37541 D08BFU 5282102 Ki = 423.7 nM T37541 D09JPC 16402 Ki = 440 nM T37541 D09LWR 3433937 Ki = 5.5 nM T37541 D09PWX 8739 Ki = 52 nM T37541 D09TES 44395768 Ki = 7.1 nM T37541 D09WSJ 19772348 Ki = 88.9 nM T37541 D09WVV 8111 Ki = 12100 nM T37541 D0A0YX 5143 Ki = 10 nM T37541 D0A1CM 5281855 Ki = 6320 nM T37541 D0A3JR 3051968 Ki = 6.9 nM T37541 D0A8HW 44395685 Ki = 1.5 nM T37541 D0AU0M 637542 Ki = 5230 nM T37541 D0C4QB 44395769 Ki = 8 nM T37541 D0C7LR 313 Ki = 1840000 nM T37541 D0D4OV 20043772 Ki = 79.6 nM T37541 D0D5XC 101753 Ki = 36150000 nM T37541 D0D6UR 12394434 Ki = 3700 nM T37541 D0E0RW 69894 Ki = 23800 nM T37541 D0E8CC 18794 Ki = 0.45 nM T37541 D0EJ9B 66827 Ki = 8300 nM T37541 D0G0FJ 11206245 Ki = 68 nM T37541 D0G3BI 25090 Ki = 32 nM T37541 D0G3TK 5280863 Ki = 25 nM T37541 D0G9NE 11659798 Ki = 8.2 nM T37541 D0H3NS 10752 Ki = 6200 nM T37541 D0HN0R 11623958 Ki = 0.78 nM T37541 D0IB3K 5320686 Ki = 4.6 nM T37541 D0J3SP 11718391 Ki = 6.8 nM T37541 D0KZ2D 11638641 Ki = 1.7 nM T37541 D0L5TZ 20195365 Ki = 17100 nM T37541 D0LC0F 96876 Ki = 5.1 nM T37541 D0LU4S 156219 Ki = 4100 nM T37541 D0M3PO 69561 Ki = 100 nM T37541 D0M6RM 7365 Ki = 12500 nM T37541 D0N1AW 45485270 Ki = 9000 nM T37541 D0N7WP 44520903 Ki = 7.7 nM T37541 D0NN3Q 78105 Ki = 89 nM T37541 D0O0UE 729977 Ki = 4.7 nM T37541 D0O4KL 11640067 Ki = 1.9 nM T37541 D0O8WV 11536481 Ki = 4.5 nM T37541 D0O9VU 44520901 Ki = 5.4 nM T37541 D0OI1H 72894 Ki = 45 nM T37541 D0OT5L 1631814 Ki = 7100 nM T37541 D0P6AM 3526523 Ki = 61 nM T37541 D0Q7DJ 10742 Ki = 7810 nM T37541 D0RB0D 44268050 Ki = 30100 nM T37541 D0S9YX 5280373 Ki = 371.5 nM T37541 D0SF3B 11529486 Ki = 6.5 nM T37541 D0SY2M 5281708 Ki = 4.2 nM T37541 D0T3NP 7456 Ki = 780 nM T37541 D0TY8X 31036 Ki = 6.8 nM T37541 D0U4BB 10748 Ki = 2400 nM T37541 D0V9EN 689043 Ki = 6420 nM T37541 D0VD7H 84724 Ki = 5.2 nM T37541 D0W1OR 7424 Ki = 7170 nM T37541 D0W9VC 670143 Ki = 6.2 nM T37541 D0X5HL 15107 Ki = 360 nM T37541 D0X6IE 4422372 Ki = 5.6 nM T37541 D0XL5K 67944 Ki = 4 nM T37541 D0Y3TZ 370 Ki = 6070 nM T37541 D0Y7HG 5281616 Ki = 24.5 nM T37541 D0YU8J 1502014 Ki = 120 nM T37541 D0Z1HY 67136 Ki = 210 nM T37541 D0Z5GE 44520902 Ki = 5.3 nM T37541 D0ZC3W 6269 Ki = 88 nM T59626 D09JUG 60490 IC50 = 420 nM T59626 D0O4NR 5280492 Ki = 0.12 nM T59626 D0S0WN 114999 IC50 = 1 nM T59626 D0DK4I 4534 IC50 = 85 nM T59626 D0NS6I 10037501 Ki = 100000 nM T59626 D00GNK 177941 Ki = 25 nM T59626 D01XMO 192617 Ki = 0.04 nM T59626 D04JJE 132425 IC50 = 60 nM T59626 D05LYL 196905 IC50 = 1.5 nM T59626 D09LQP 132379 Ki = 0.14 nM T59626 D0B6JV 6435820 Ki = 7.1 nM T59626 D0C0EO 9867257 IC50 = 8.4 nM T59626 D0G7SP 6441619 Ki = 0.78 nM T59626 D0JY4Y 443292 IC50 = 210 nM T59626 D0NK8D 204058 Ki = 1.3 nM T59626 D0OP7B 6450158 Ki = 5.9 nM T59626 D0U9JL 6444688 IC50 = 1.9 nM T59626 D0Y2IH 122023 Ki = 77 nM T59626 D0Z0OT 6438358 Ki = 3.7 nM T59626 D0Z1TF 9850974 Ki = 1 nM T59626 CPVH47 129065 IC50 = 30 nM T59626 CY35ZC 178581 IC50 = 20 nM T59626 C6E7UC 192624 Ki = 3.467 nM T59626 C2DP3F 195214 IC50 = 210 nM T59626 C4JBN5 204055 IC50 = 3.2 nM T59626 CLJ1V0 3083459 Ki = 4.677 nM T59626 CLG18V 6439436 Ki = 4.7 nM T59626 CBM47Q 6852392 Ki = 700 nM T59626 COF3U8 9800998 Ki = 38000 nM T59626 CQ94JS 9805394 IC50 = 2.4 nM T59626 CVP13O 9807782 Ki = 4 nM T59626 C92QAN 9826485 Ki = 280 nM T59626 CS4D7L 9829619 Ki = 14 nM T59626 C4GI1E 9845585 Ki = 33.88 nM T59626 CF04AP 9845587 Ki = 61.66 nM T59626 CM76TV 9849151 IC50 = 610 nM T59626 CRS48K 9850643 Ki = 1 nM T59626 CVP79S 9865985 IC50 = 1 nM T59626 C78PTA 9872540 Ki = 42 nM T59626 CMGA15 9911868 IC50 = 7 nM T59626 CF7Y2J 9912012 Ki = 3.51 nM T59626 C67CBX 9930128 IC50 = 15.9 nM T59626 C5NBC4 9934323 IC50 = 43 nM T59626 CX38IE 9934500 IC50 = 800 nM T59626 CJSG78 9955657 IC50 = 4 nM T59626 CHY6Q3 9958441 Ki = 1.5 nM T59626 CFP2X1 9959228 Ki = 80 nM T59626 CLH47O 9976757 IC50 = 4 nM T59626 C0JM4I 9976891 IC50 = 8000 nM T59626 CHV5W2 9978895 IC50 = 6 nM T59626 CKLU93 9980059 IC50 = 1200 nM T59626 CDN4R5 9984593 Ki = 15.4 nM T59626 CGJ5W3 9985159 IC50 = 1150 nM T59626 C2JAZ3 9999718 IC50 = 40 nM T59626 CZ21UT 9999755 IC50 = 10 nM T59626 CI9NV6 10001576 IC50 = 5 nM T59626 CPJ5S8 10007005 IC50 = 25 nM T59626 CHF5J3 10019853 IC50 = 700 nM T59626 CH4U8L 10021622 IC50 = 2000 nM T59626 CV2HL3 10022413 IC50 = 45 nM T59626 CGL59Z 10023244 IC50 = 5 nM T59626 CCT4B7 10024190 IC50 = 110 nM T59626 CZ79EA 10032156 IC50 = 5800 nM T59626 CPUH04 10046386 IC50 = 2500 nM T59626 CC18QV 10046878 IC50 = 4 nM T59626 CYFS74 10047140 IC50 = 5 nM T59626 CFGB01 10050724 Ki = 4.8 nM T59626 C1CZP6 10052488 IC50 = 1100 nM T59626 COIH64 10052575 IC50 = 93 nM T59626 C8S0KE 10053028 IC50 = 320 nM T59626 CH5J9D 10053662 IC50 = 12.3 nM T59626 CD1O6X 10068808 IC50 = 400 nM T59626 C9CP2E 10069416 IC50 = 15 nM T59626 CNW4B1 10069417 IC50 = 1100 nM T59626 CIQS13 10071290 IC50 = 10000 nM T59626 CD7AP1 10090758 IC50 = 40 nM T59626 C85COL 10091738 IC50 = 13 nM T59626 CR45PL 10092630 IC50 = 9.5 nM T59626 C4A1IL 10120811 Ki = 0.14 nM T59626 CK4UL8 10159791 Ki = 58.88 nM T59626 C0K3FJ 10179915 Ki = 3.02 nM T59626 C5DH9M 10182429 Ki = 20.42 nM T59626 CI8DY3 10247237 IC50 = 550 nM T59626 CQ2R1G 10248148 IC50 = 183 nM T59626 COX86A 10250881 IC50 = 150 nM T59626 C7IR8W 10257351 Ki = 8 nM T59626 C73LQM 10314767 IC50 = 300 nM T59626 CK0W8I 10315808 IC50 = 1800 nM T59626 CYK46J 10318241 IC50 = 5 nM T59626 C1B8HI 10319829 IC50 = 22 nM T59626 C7XK2U 10324028 Ki = 28 nM T59626 CAES31 10325873 Ki = 240 nM T59626 CC1UF0 10335738 IC50 < 100 nM T59626 CFHI60 10337448 IC50 = 700 nM T59626 CHU5F0 10339300 IC50 = 68.2 nM T59626 C5X4IP 10340408 IC50 = 500 nM T59626 CMR45D 10341135 IC50 = 50 nM T59626 CV1KW5 10341242 IC50 = 2 nM T59626 CC3VK8 10342316 Ki = 38.02 nM T59626 CKH19Z 10343923 IC50 = 2 nM T59626 CB58OJ 10346127 Ki = 9.2 nM T59626 CCYB57 10347709 IC50 = 890 nM T59626 CH71MO 10349070 IC50 = 750 nM T59626 CQZ6S3 10362331 IC50 = 30 nM T59626 C2UW4Y 10363485 Ki = 38000 nM T59626 CP7IQ1 10363959 IC50 = 600 nM T59626 CZIL76 10364772 IC50 = 4.2 nM T59626 C6FS8B 10371282 Ki = 53 nM T59626 C5XYM3 10385899 IC50 = 10 nM T59626 CF9RH8 10386030 IC50 = 200 nM T59626 C2X5KM 10387303 IC50 = 300 nM T59626 CR9Q0B 10387480 IC50 = 30 nM T59626 CN1KZ9 10390056 IC50 = 150 nM T59626 C6M8ZS 10391552 IC50 = 520 nM T59626 CD05VJ 10406292 IC50 = 3 nM T59626 C2SCY7 10407131 IC50 = 300 nM T59626 CN0WY3 10407251 IC50 = 100 nM T59626 CZ1PY3 10415106 IC50 = 44500 nM T59626 C25MYB 10425738 IC50 < 100 nM T59626 C6V2ZW 10427789 IC50 = 50 nM T59626 C2PRE8 10430674 IC50 = 18 nM T59626 CJM40K 10430678 IC50 = 300 nM T59626 C2DHB5 10430946 IC50 = 2000 nM T59626 C8G7SN 10436331 IC50 = 5.2 nM T59626 C1HD2M 10451768 IC50 = 30 nM T59626 CE5VO0 10455429 IC50 = 300 nM T59626 C59MAC 10474073 IC50 > 1000 nM T59626 C5CQU8 10474602 IC50 = 15 nM T59626 C16TRD 10475503 IC50 = 5 nM T59626 C0CD8E 10475982 Ki = 16000 nM T59626 CU7FJ6 10477988 IC50 = 20 nM T59626 C6OV4L 10481412 IC50 = 770 nM T59626 C7WUL1 10482767 IC50 = 26 nM T59626 CQ23JE 10483151 IC50 = 2800 nM T59626 CWS3I5 10507666 Ki = 36 nM T59626 CK9MR2 10529082 Ki = 1.2 nM T59626 CK1X4N 10529241 Ki = 1.3 nM T59626 CJ9OI2 10554820 Ki = 33 nM T59626 CS65WD 10600128 Ki = 66.07 nM T59626 CEYL09 10625086 IC50 > 300 nM T59626 CH3FV2 10648186 Ki = 1.4 nM T59626 CSAF60 10670634 Ki = 63.1 nM T59626 CQ4S9P 10692884 Ki = 9.5 nM T59626 C3YMX7 10694814 Ki = 2.8 nM T59626 C5FXV6 10737187 IC50 = 900 nM T59626 CGT19D 10741106 IC50 = 80 nM T59626 C35FCG 10745069 Ki = 25 nM T59626 C35LWJ 10745838 Ki = 0.11 nM T59626 CMV5O6 10793277 Ki = 5.9 nM T59626 CO36IA 10812265 Ki = 16.22 nM T59626 CKH76L 11725988 IC50 = 500 nM T59626 C5WMJ9 11726048 IC50 = 150 nM T59626 CRDS63 11740566 IC50 = 800 nM T59626 CAO1X6 11741184 IC50 = 1000 nM T59626 CJP4L1 11756030 IC50 = 100 nM T59626 C24LXS 11798329 Ki = 12 nM T59626 CG1TE6 11798848 Ki = 1.5 nM T59626 C4EZ9M 11799000 IC50 = 60 nM T59626 CSR1I5 11800543 Ki = 12 nM T59626 C7HA8C 14282627 IC50 = 26200000 nM T59626 CS8T7E 14946858 IC50 = 100 nM T59626 C5MO7U 14977894 Ki = 429 nM T59626 CRH1W3 14977898 Ki = 165 nM T59626 C8VTF9 14977907 Ki = 1130 nM T59626 C1G0DR 14977911 Ki = 338 nM T59626 CK6B9V 14977913 Ki = 150 nM T59626 CWNE34 14977916 Ki = 478 nM T59626 C4WAQ7 14977920 Ki = 252 nM T59626 C76KWU 14977924 Ki = 151 nM T59626 C5IT0Y 14977927 Ki = 284 nM T59626 CZCJ15 14977931 Ki = 34 nM T59626 CL46SC 14977933 Ki = 36 nM T59626 C1VS5J 14977939 Ki = 74 nM T59626 CPR26X 14977943 Ki = 72 nM T59626 CDPY62 14977946 Ki = 148 nM T59626 CT59OE 14977948 Ki = 609 nM T59626 CC42FK 14977952 Ki = 147 nM T59626 CV70FZ 14977955 Ki = 789 nM T59626 C8RJ2H 14977957 Ki = 36 nM T59626 C81AXN 14977959 Ki = 11 nM T59626 C45IKJ 14977961 Ki = 43 nM T59626 C73MEH 14977963 Ki = 14 nM T59626 CPQ5E3 14977965 Ki = 12 nM T59626 CK79ZP 15227776 Ki = 3.53 nM T59626 C8JPS3 15658097 Ki = 900 nM T59626 CAX32C 15658098 Ki = 1400 nM T59626 CRZV56 15658099 Ki = 2800 nM T59626 CJ5R9F 15658119 Ki = 600 nM T59626 C80ROL 15658122 Ki = 140 nM T59626 CT83ZJ 15658147 Ki = 1 nM T59626 C2KPE8 15666575 IC50 = 10000 nM T59626 CH1QG8 15666577 IC50 = 1000 nM T59626 C5Z7NC 15666578 IC50 = 1000 nM T59626 C9FEK1 15666579 IC50 = 1000 nM T59626 CT4IA8 15666581 IC50 = 5000 nM T59626 C1EG6H 15666582 IC50 = 3000 nM T59626 CBC62V 15666586 IC50 = 700 nM T59626 CV67IJ 15666588 IC50 = 300 nM T59626 CEDG15 15666597 IC50 = 10000 nM T59626 C9WXO4 15666601 IC50 = 3500 nM T59626 C83QOF 15666603 IC50 = 1000 nM T59626 CH07PD 15666610 IC50 = 4500 nM T59626 C2CSJ4 15666613 IC50 = 1500 nM T59626 C9BL8Z 15666614 IC50 = 300 nM T59626 CFQ59K 15666615 IC50 = 200 nM T59626 CX1UQ4 15666618 IC50 = 110 nM T59626 CL86KV 15666621 IC50 = 1000 nM T59626 C8PU5J 15666623 IC50 = 800 nM T59626 C5LOM8 15666630 IC50 = 3000 nM T59626 C3N8MR 15666631 IC50 = 6000 nM T59626 CSH98I 15718079 IC50 = 1766 nM T59626 C0R7QD 15718082 IC50 = 2097 nM T59626 CV0YI1 15718085 IC50 = 832 nM T59626 CC2ER7 15839729 IC50 = 39.6 nM T59626 CJMU02 15839731 Ki = 4.96 nM T59626 CO70YW 15839732 Ki = 18.5 nM T59626 C7T8QY 15839733 Ki = 15.5 nM T59626 CCSA24 15839735 IC50 = 190 nM T59626 C0IX4S 15839751 Ki = 1.2 nM T59626 C0HRV3 18373300 IC50 = 500 nM T59626 C5GXB8 18373357 IC50 = 400 nM T59626 CDM6Q7 18373405 IC50 = 400 nM T59626 C9HF6C 18963032 Ki = 1.93 nM T59626 C7NL1V 19600933 Ki = 0.073 nM T59626 C8W2UP 21765772 Ki = 5.7 nM T59626 CD4K3V 21765774 Ki = 161 nM T59626 CMZU98 21765776 Ki = 112 nM T59626 CIF6K8 23257866 Ki = 129 nM T59626 CTBZ01 23257882 Ki = 245 nM T59626 CG0XA7 23257889 Ki = 192 nM T59626 CRG1H3 23257891 Ki = 232 nM T59626 CE2NF8 23257894 Ki = 37 nM T59626 C3TVL7 23501721 IC50 = 0.48 nM T59626 C90URE 23672801 Ki = 100 nM T59626 C3AP9Q 23672802 Ki = 50 nM T59626 CB9CM0 23672803 Ki = 9000 nM T59626 C2V8OU 23672804 Ki = 500 nM T59626 CZM4J7 23672805 Ki = 1 nM T59626 CGW18L 23672806 Ki = 60 nM T59626 CM9FX3 23672807 Ki = 3 nM T59626 CJ34EX 23672808 Ki = 1000 nM T59626 CC6PW9 23682552 IC50 = 300 nM T59626 C3A8CU 23699208 Ki = 10.3 nM T59626 CJMZ37 25174150 IC50 = 0.07 nM T59626 CVB0H8 25191879 IC50 = 0.18 nM T59626 C3JX1S 25191880 IC50 = 0.2 nM T59626 CV3TA6 25192021 IC50 = 0.21 nM T59626 C9WI6J 25192023 IC50 = 0.22 nM T59626 C2W9JA 25192174 IC50 = 0.36 nM T59626 CGV6N8 25192175 IC50 = 0.39 nM T59626 C7E8AM 25192176 IC50 = 0.38 nM T59626 CX3P6J 25192325 IC50 = 0.57 nM T59626 CO1E8H 25192326 IC50 = 0.58 nM T59626 CC6OR8 25192327 IC50 = 0.58 nM T59626 C9UL8Y 25192468 IC50 = 0.61 nM T59626 C7A8UE 25192471 IC50 = 1.19 nM T59626 CYK6X5 44213761 IC50 = 300 nM T59626 CP1F9I 44270188 Ki = 15.4 nM T59626 CA73JM 44275225 IC50 > 2000 nM T59626 CRM07V 44290966 Ki = 65.7 nM T59626 CZ8S4B 44291011 IC50 = 6.6 nM T59626 C7VKX3 44291012 IC50 = 35.6 nM T59626 CY5Q3Z 44291013 IC50 = 30.8 nM T59626 C24UOY 44291014 IC50 = 41.5 nM T59626 CG39HS 44291030 IC50 = 12 nM T59626 CM2A0S 44291031 Ki = 4.75 nM T59626 CDO50G 44296838 IC50 = 3800 nM T59626 CRGM38 44302134 Ki = 6.8 nM T59626 CP81YA 44302954 Ki = 5.53 nM T59626 C2GA3P 44302962 Ki = 28.4 nM T59626 C07QMJ 44302965 Ki = 3.2 nM T59626 C3MJH6 44302966 Ki = 320 nM T59626 CGQ38X 44302971 Ki = 5.14 nM T59626 C9XI2B 44302983 Ki = 6.51 nM T59626 CLT39P 44315538 IC50 = 70000 nM T59626 CE06WF 44315582 IC50 = 8000 nM T59626 CFU18I 44315784 IC50 = 1000 nM T59626 CQ0U2I 44317392 IC50 = 319 nM T59626 CAIE35 44337707 IC50 = 1200 nM T59626 CKL2R3 44340786 Ki = 10 nM T59626 C5E9JY 44341073 Ki = 27000 nM T59626 CY3XG6 44341107 Ki = 19000 nM T59626 CXJ7K3 44341141 Ki = 225 nM T59626 C1JQ9S 44341265 Ki = 9000 nM T59626 C1QIP7 44341318 Ki = 2400 nM T59626 CA39XW 44348541 IC50 = 50 nM T59626 CS9G0A 44356239 IC50 = 4700 nM T59626 C35ENC 44357534 IC50 = 50 nM T59626 C2S4FU 44357546 IC50 = 7 nM T59626 CLIK19 44359651 IC50 = 400 nM T59626 CE5Z1Q 44379572 IC50 = 6000 nM T59626 CS7I2Y 44379573 IC50 = 2000 nM T59626 C6PUO7 44379592 IC50 = 2000 nM T59626 CI2VA5 44379910 IC50 > 10000 nM T59626 C3JC5B 44381856 IC50 = 15.5 nM T59626 CL8B3S 44382275 Ki = 330 nM T59626 C4HZU0 44382276 Ki = 5200 nM T59626 C4N9UJ 44382378 IC50 = 220 nM T59626 CU8SD4 44382384 Ki = 3300 nM T59626 CEU1A0 44382463 Ki = 39000 nM T59626 C05WVE 44382468 Ki = 1900 nM T59626 CAOW45 44384957 IC50 = 784 nM T59626 CJT8L2 44384958 IC50 = 276 nM T59626 C93RQX 44385131 IC50 = 1180 nM T59626 CQ3AK6 44385159 IC50 = 1220 nM T59626 C8Y5RF 44385160 IC50 = 4570 nM T59626 C4M3OJ 44385199 IC50 = 1510 nM T59626 C1TZE0 44385218 IC50 = 1180 nM T59626 CA9FK0 44385257 IC50 > 10000 nM T59626 CQ5HY6 44385258 IC50 = 190 nM T59626 CAT57Z 44385920 IC50 = 830 nM T59626 CJQM34 44385966 IC50 = 932 nM T59626 C7X2YA 44386171 IC50 = 908 nM T59626 CRDA84 44386172 IC50 = 16.7 nM T59626 COL05K 46888195 IC50 = 8.5 nM T59626 CK20OJ 46888196 IC50 = 31.1 nM T59626 CXNZ90 46888197 IC50 = 5.35 nM T59626 CLK29W 46888198 IC50 = 5.39 nM T59626 C24FWR 46888199 IC50 = 139.7 nM T59626 C5A4PJ 46888200 IC50 = 13.98 nM T59626 C3BSZ4 46888201 IC50 = 3.27 nM T59626 CS6CR7 46888202 IC50 = 60.2 nM T59626 C62DUR 135401173 IC50 = 12 nM T59626 C8GIO2 135430350 IC50 = 738 nM T59626 C8YS2G 135457469 IC50 = 9.3 nM T59626 CV6YJ0 135500104 IC50 = 87 nM T59626 C1GON6 135503765 IC50 = 11 nM T59626 C1A9MF 135507183 IC50 = 54 nM T59626 C72JDF 135507225 IC50 = 55 nM T59626 CVB8W3 135507252 IC50 = 28 nM T59626 C84SWJ 135507273 IC50 = 834 nM T59626 C4V2EX 135516891 IC50 = 6.4 nM T59626 CCSR81 135531245 IC50 = 107 nM T59626 C6WFG1 135543741 IC50 = 82 nM T59626 C7MEH5 135543742 IC50 = 5.7 nM T59626 C4XA8E 135543808 IC50 = 4.5 nM T59626 D00HYO 20704716 Ki = 5300 nM T59626 D05HNB 9893718 Ki = 1.2 nM T59626 D06IJI 44379678 IC50 = 0.1 nM T59626 D07EGC 15817161 IC50 = 0.85 nM T59626 D09QJS 9958915 IC50 = 8.5 nM T59626 D0C2GW 44379453 IC50 = 0.15 nM T59626 D0F4EL 10021742 Ki = 1300 nM T59626 D0H6YL 44403368 IC50 = 8 nM T59626 D0L8VT 44403823 IC50 = 54 nM T59626 D0R9ED 15237280 IC50 = 5.3 nM T59626 D0V3ZG 25192022 IC50 = 114 nM T59626 D0ZB8S 44379679 IC50 < 0.1 nM T15571 D01AZG 5073 Ki = 1000 nM T15571 D01TSI 8223 Ki = 14 nM T15571 D03WEX 9966051 Ki = 220 nM T15571 D08VRO 3822 Ki = 20000 nM T15571 D0CQ0Z 33630 Ki = 1000 nM T15571 D0G8NN 119570 Ki > 10000 nM T15571 D0H3HM 60795 Ki = 1000 nM T15571 D0H7KF 5002 Ki > 1000 nM T15571 D0V4QS 135398745 Ki > 1000 nM T15571 D0W5HK 216239 Ki = 3296 nM T15571 D0Z1RV 135398737 Ki = 1000 nM T15571 D0Z6UC 5358 IC50 = 501.19 nM T15571 D0N1HW 5311200 Ki > 10000 nM T15571 D00OWF 5280953 Ki > 10000 nM T15571 D08AWI 11430856 Ki > 5000 nM T15571 D0M7LV 5761 Ki = 9 nM T15571 D0YP7L 6604889 Ki = 63.1 nM T15571 CUQ05A 3564 Ki > 10000 nM T15571 C2QLD4 3565 Ki > 10000 nM T15571 C5H9CN 9287 Ki > 10000 nM T15571 C6WDL7 49756 Ki = 10450 nM T15571 CHKO01 91522 Ki > 10000 nM T15571 CX1GC4 108182 Ki = 16000 nM T15571 CP9D2L 151142 Ki < 10 nM T15571 C6RSI8 159809 Ki > 10000 nM T15571 CGT8R0 160510 Ki = 845 nM T15571 CYV1R3 417052 Ki > 10000 nM T15571 CAH9F5 656705 Ki > 10000 nM T15571 C2VLP8 752521 Ki = 389 nM T15571 COG8R1 2058916 Ki > 10000 nM T15571 CA2OY6 2737389 Ki = 76 nM T15571 CS8KE2 3649661 Ki = 457 nM T15571 C6SHA4 4713248 Ki = 5000 nM T15571 C8HQN1 5376026 Ki > 10000 nM T15571 C3MA1N 9819150 IC50 = 794.33 nM T15571 CM13ZV 9856041 Ki > 10000 nM T15571 CJW1P5 9888494 Ki = 1479.11 nM T15571 CUN81Q 9905249 Ki > 10000 nM T15571 CYWQ50 9906447 Ki > 10000 nM T15571 CWC69L 9998879 IC50 = 501.19 nM T15571 CV7R9F 10020040 Ki > 10000 nM T15571 C86UFO 10021702 IC50 = 125.89 nM T15571 C2EUY0 10035109 Ki > 10000 nM T15571 C92UGJ 10043491 IC50 = 125.89 nM T15571 CH25VX 10245588 IC50 = 630.96 nM T15571 CH31DX 10267394 Ki > 10000 nM T15571 CU89JD 10314060 Ki > 10000 nM T15571 CAS0N1 10315894 IC50 = 199.53 nM T15571 C7M5TZ 10337965 IC50 = 251.19 nM T15571 C6C3HX 10340828 IC50 = 79.43 nM T15571 C8FB4S 10382508 Ki = 13 nM T15571 CP3OG2 10383252 IC50 = 1000 nM T15571 C9MXP8 10404070 IC50 = 1995.26 nM T15571 CHD23R 10404770 IC50 = 125.89 nM T15571 CYM5R8 10412397 IC50 = 199.53 nM T15571 C2B0IU 10421236 IC50 > 10000 nM T15571 C5RH4N 10471382 IC50 = 794.33 nM T15571 CY0EK4 10471383 IC50 = 794.33 nM T15571 COV85C 10472143 Ki = 27 nM T15571 CP8WN3 10872812 Ki = 200 nM T15571 CXP8H3 10881882 Ki = 930 nM T15571 CI9Z8E 10882775 Ki = 200 nM T15571 CRI50E 10885636 IC50 = 3380 nM T15571 CGI03V 10893866 Ki = 250 nM T15571 C1BF4J 10924201 Ki = 1920 nM T15571 CXFH06 10926167 Ki = 350 nM T15571 CNB39C 10947658 Ki = 16 nM T15571 C3X5OI 11035049 Ki = 190 nM T15571 C3AJ7L 11074351 Ki > 10000 nM T15571 CM9KX0 11088692 Ki = 1080 nM T15571 CVE8T3 11121216 Ki = 13 nM T15571 CS3YK5 11352884 Ki = 25.12 nM T15571 CF1O2M 11364267 Ki = 31.62 nM T15571 C85LYP 11430418 IC50 > 1000 nM T15571 C5C6ZJ 11443218 Ki = 125.89 nM T15571 CNH1K4 11568826 Ki > 10 nM T15571 CGX8F6 11596869 Ki > 6900000 nM T15571 C4L7TV 11662592 Ki > 1 nM T15571 C9X7EK 11722814 IC50 = 630.96 nM T15571 CE5C1J 11726973 Ki = 620 nM T15571 C7PVL8 11730467 IC50 = 5520 nM T15571 C7X4KL 11759441 Ki > 10000 nM T15571 CO9YM4 11808247 Ki = 400 nM T15571 CXLW54 11948707 Ki > 10000 nM T15571 C8JQL7 11957735 IC50 > 10000 nM T15571 C20RFT 14935215 Ki > 10000 nM T15571 C7VAI1 15011772 IC50 > 10000 nM T15571 C1LWZ6 16006605 Ki = 6.5 nM T15571 CK36NS 16006607 Ki = 10 nM T15571 CD3E8L 16093484 Ki = 2 nM T15571 CEW91O 16093485 Ki = 4.7 nM T15571 CZ2IS9 16660294 Ki > 10000 nM T15571 C7T8JC 19958494 Ki > 10000 nM T15571 C6LI5E 19958507 Ki > 10000 nM T15571 C3T5HF 21509921 Ki = 741.31 nM T15571 CT7XG9 21830793 Ki > 10000 nM T15571 CBN84K 22065997 Ki > 10000 nM T15571 CZ7J4B 22857296 Ki = 630 nM T15571 CDC91N 24839550 Ki < 10000 nM T15571 CY21RE 24841480 Ki = 2200 nM T15571 C3HK0J 24865725 Ki = 1258.93 nM T15571 C0O6FX 24865727 Ki = 1584.89 nM T15571 CUY89J 24936155 Ki = 3000 nM T15571 CJ3NP5 42636941 IC50 > 10000 nM T15571 CCP07F 44275750 Ki = 3 nM T15571 CC2OD4 44278111 Ki > 10000 nM T15571 CRMA84 44278114 Ki > 10000 nM T15571 CF0Y4M 44278115 Ki > 10000 nM T15571 CER86D 44327952 Ki = 200 nM T15571 CN3QX1 44351063 Ki = 1775 nM T15571 C57PAS 44351077 Ki = 285 nM T15571 C4WY3Z 44351100 Ki = 185 nM T15571 CR85QU 44351102 Ki = 174 nM T15571 CI47MT 44351116 Ki = 1120 nM T15571 C2J6RG 44351139 Ki = 100 nM T15571 CTF6U8 44351140 Ki = 100 nM T15571 CD1JZ2 44351180 Ki = 225 nM T15571 CP92MG 44351183 Ki = 1395 nM T15571 C7H6ZS 44351184 Ki = 165 nM T15571 CSW4B9 44351193 Ki = 270 nM T15571 CYO3S8 44351342 Ki = 168 nM T15571 CD5E1G 44374431 Ki = 287 nM T15571 CK28HY 44374637 Ki > 3448 nM T15571 C8EK9X 44374648 Ki = 3067 nM T15571 CA0W9E 44397360 Ki = 31.62 nM T15571 CL96VK 44397361 Ki = 79.43 nM T15571 C7YV9X 44397363 Ki = 25.12 nM T15571 C1AVF4 44397364 Ki = 5.012 nM T15571 CE2ZW4 44397426 Ki = 501.19 nM T15571 CO8J2L 44397428 Ki = 6309.57 nM T15571 CD85BN 44397430 Ki = 1000 nM T15571 CK7DX8 44397432 Ki = 630.96 nM T15571 CJ1UF5 44397434 Ki = 398.11 nM T15571 CS2E6D 44397486 Ki = 199.53 nM T15571 CODE60 44397510 Ki = 3162.28 nM T15571 C4K0MN 44397512 Ki = 251.19 nM T15571 C4B0OI 44397588 Ki = 25.12 nM T15571 C5FP0R 44397589 Ki = 50.12 nM T15571 C6GSJ1 44397592 Ki = 251.19 nM T15571 CYJF09 44397618 Ki = 12.59 nM T15571 C2AGC5 44397667 Ki = 199.53 nM T15571 CA46QM 44397668 Ki = 79.43 nM T15571 CE3G8U 44397670 Ki = 6.31 nM T15571 CG87PW 44409290 Ki > 720 nM T15571 CZL97F 44455426 Ki > 10000 nM T15571 CYS7T4 44455943 Ki = 26.5 nM T15571 CPJ16W 44455962 Ki = 415 nM T15571 CO7TM5 44455963 Ki = 122 nM T15571 C4DAW2 44455980 Ki = 1172 nM T15571 CGBA20 44455982 Ki > 10000 nM T15571 CY7B1J 44455985 Ki = 38 nM T15571 C6BFI0 44456033 Ki = 1.6 nM T15571 CCE8Z7 44456170 Ki = 1990 nM T15571 CBU1G5 44456207 Ki = 97 nM T15571 CTF4X6 44456246 Ki = 463 nM T15571 C5SYI3 44456251 Ki = 1375 nM T15571 C45ELH 44456253 Ki = 647 nM T15571 C1WX4S 44456284 Ki = 274 nM T15571 CB34EP 44456286 Ki = 911 nM T15571 CG91RD 44456395 Ki = 22.9 nM T15571 C4X0ZV 44456398 Ki = 882 nM T15571 C12XGE 44456400 Ki = 466 nM T15571 CYUQ72 44456443 Ki = 550 nM T15571 C6NE3T 44456487 Ki = 145 nM T15571 C4DL5C 44469677 IC50 = 1 nM T15571 CRCH48 44582675 Ki = 6814 nM T15571 CEJ4R8 44582676 Ki = 1584 nM T15571 CZGP86 44582677 Ki > 10000 nM T15571 C5QB4K 44582678 Ki > 10000 nM T15571 C01RCI 44582705 Ki = 1684 nM T15571 CXL25V 44582706 Ki > 10000 nM T15571 C8MR1X 44582707 Ki > 10000 nM T15571 C4IT1N 44582708 Ki > 10000 nM T15571 CVJ04W 45263888 Ki = 99 nM T15571 CZOG43 45266001 Ki = 347 nM T15571 C2LZJ0 49783209 Ki = 8589 nM T15571 C57SMG 49783415 Ki > 10000 nM T15571 C0TG6I 49783419 Ki > 10000 nM T15571 CR40BA 49836386 IC50 > 1000 nM T15571 C2RY0J 50878551 Ki = 3311.31 nM T15571 C1W6TV 50898777 Ki > 10000 nM T15571 CXMZ73 50898778 Ki > 10000 nM T15571 CE4KP1 51050257 Ki > 10000 nM T15571 CRQF15 53325242 Ki = 894 nM T15571 CG24AT 53381002 Ki = 1525 nM T15571 CH37LU 56663451 IC50 > 10000 nM T15571 C1TC7Q 56963799 Ki > 10000 nM T15571 C1LEH8 67268994 Ki > 10000 nM T15571 C3XNC2 71450247 Ki > 10000 nM T15571 C9VZ8J 71450550 Ki > 10000 nM T15571 CYK20Z 71452384 Ki > 10000 nM T15571 C7UCP8 71452650 Ki = 208 nM T15571 CAQF34 71455625 Ki > 10000 nM T15571 CMJ1O9 71457409 Ki > 10000 nM T15571 CS83IF 71459269 Ki = 1700 nM T15571 CK5T4P 71459604 Ki = 7815 nM T15571 C63YLA 71461049 Ki > 10000 nM T15571 CJD96I 71461050 Ki > 10000 nM T15571 C4P3JU 71462776 Ki = 5805 nM T15571 C3GUQ2 71462777 Ki > 10000 nM T15571 CWH6T3 72548703 IC50 = 106 nM T15571 C8Z0NM 72550642 Ki = 1178 nM T15571 CL6W2Q 72550645 Ki = 517 nM T15571 C78LYM 72698087 Ki > 10000 nM T15571 C63HPK 72698088 Ki > 10000 nM T15571 CC6Q5R 72771081 Ki < 100 nM T15571 CC65OA 73213195 Ki > 10000 nM T15571 CW83DK 73213196 Ki > 10000 nM T15571 CCV91B 73346042 Ki = 2128 nM T15571 C1NJ0R 73353884 Ki = 6060 nM T15571 C4F7VK 73355415 Ki = 7502 nM T15571 C2E7QW 75201901 Ki > 10000 nM T15571 C8IDL3 75306277 Ki = 199.53 nM T15571 CEMZ15 118464420 Ki = 227 nM T15571 CV2L6O 118464425 Ki = 595 nM T15571 CFNG86 118464427 Ki = 994 nM T15571 CLW53P 122483274 Ki = 337 nM T15571 CO63ET 122483280 Ki = 5 nM T15571 C4QM2E 124247485 Ki > 10000 nM T15571 CTBN56 127026052 Ki = 4265.8 nM T15571 C0SZI4 127026515 Ki = 933 nM T15571 CU49VE 127036186 Ki = 3235.94 nM T15571 CG06BD 127036932 Ki = 2089.3 nM T15571 CVW71O 127036953 Ki = 2398.83 nM T15571 C50GOC 130442480 Ki = 9500 nM T15571 CM04RF 130442572 Ki = 7400 nM T15571 C1RI8Q 132060720 Ki = 875 nM T15571 CGHO19 132060770 Ki > 10000 nM T15571 CT81OY 132060776 Ki = 1747 nM T15571 CAVB41 132584404 Ki > 10000 nM T15571 CBU81N 134149168 Ki > 10000 nM T15571 C6N8GM 135367405 Ki > 10000 nM T15571 C6LU0C 135367816 Ki > 10000 nM T15571 CD2TH9 135367820 Ki = 1231 nM T15571 C5AMD9 135367857 Ki = 1135 nM T15571 CVE08Y 135458392 Ki = 10.72 nM T15571 CP7HN4 135458393 Ki = 6.31 nM T15571 CS8XJ6 135458394 Ki = 6.3 nM T15571 C9B7XA 135458410 Ki = 5.7 nM T15571 CFV9A3 135458427 Ki = 22.2 nM T15571 CKX4N8 135458428 Ki = 28.2 nM T15571 CTE23K 135464118 Ki = 89 nM T15571 C7AGR0 135474338 Ki = 5355 nM T15571 C1CZ9M 135514796 Ki = 101 nM T15571 CA1M8B 135966709 Ki = 25.4 nM T15571 CUKO20 136020617 Ki > 10000 nM T15571 COF0U5 136020618 Ki > 10 nM T15571 CF89JI 136030596 Ki > 10000 nM T15571 CE8GB9 136030693 Ki > 10000 nM T15571 C65VFI 136030744 Ki > 10000 nM T15571 COIX80 136054961 Ki > 10000 nM T15571 C7JHO0 136100333 Ki = 1791 nM T15571 C19GLK 136116062 Ki = 33.4 nM T15571 CA3JC8 136118613 Ki = 1282 nM T15571 CQ2GP6 136118614 Ki = 2332 nM T15571 C6R4IC 136118615 Ki = 1550 nM T15571 CS0JL5 136118616 Ki = 1454 nM T15571 CHWC38 136118619 Ki = 1425 nM T15571 C5UDW3 136118620 Ki = 7828 nM T15571 CLH0V9 136118648 Ki = 3372 nM T15571 CR72MQ 136118651 Ki = 3324 nM T15571 C0W1TM 136118658 Ki = 5080 nM T15571 C40LYH 136118659 Ki = 9118 nM T15571 CZ7C3Y 136118660 Ki = 4681 nM T15571 C42FCS 136118661 Ki = 6913 nM T15571 CR3DK1 136118716 Ki = 123 nM T15571 CON04G 136118728 Ki = 184 nM T15571 COX1F8 136118729 Ki = 112 nM T15571 C0R5PV 136118732 Ki = 1323 nM T15571 CB7N0X 136152962 Ki = 103 nM T15571 C01THU 136152963 Ki = 1472 nM T15571 CB12QP 136152964 Ki = 6.8 nM T15571 CRK8C7 136152965 Ki = 124 nM T15571 CFX06E 136152966 Ki = 22.2 nM T15571 C1UKM5 136152967 Ki = 96 nM T15571 CX0R8L 136152968 Ki = 163 nM T15571 CB8A6N 136152969 Ki = 279 nM T15571 C1JQG9 136152970 Ki = 37 nM T15571 C37YXA 136152971 Ki = 1.8 nM T15571 CY0C1X 136152972 Ki = 504 nM T15571 CFQR93 136152973 Ki = 241 nM T15571 CTW8Y5 136152974 Ki = 176 nM T15571 C0WP1E 136152976 Ki = 488 nM T15571 CQXB23 136152977 Ki = 87 nM T15571 CD81KX 136152978 Ki = 397 nM T15571 CP2M7N 136152980 Ki = 189 nM T15571 C26MKZ 136152981 Ki = 153 nM T15571 C90OMK 136179599 Ki = 196 nM T15571 CAE39V 136188797 Ki > 10000 nM T15571 CLAP52 136259032 Ki > 10000 nM T15571 C7KC3T 145963830 Ki = 4700 nM T15571 CHDN35 145964150 Ki > 10000 nM T15571 C1KH2E 145964159 Ki > 10000 nM T15571 C12OVL 145965034 Ki > 10000 nM T15571 C5W4LM 145965940 Ki > 10000 nM T15571 C81VUO 145967771 Ki > 10 nM T15571 CJS56K 145967795 Ki = 8200 nM T15571 CQJ5O8 145971635 Ki > 10000 nM T15571 C79TNE 145972796 Ki > 10000 nM T15571 C6XIN0 145974114 Ki > 10000 nM T15571 CD8ZL6 145974750 Ki > 10 nM T15571 C6PH4F 145975226 Ki > 10000 nM T15571 C71CYU 145975946 Ki > 10000 nM T15571 C2TN8W 145976085 Ki > 10000 nM T15571 C6BFY7 145977338 Ki > 10000 nM T15571 C0Y6QO 145977799 Ki = 6800 nM T15571 C3BI1R 145978113 Ki > 10000 nM T15571 CQU8R0 145978665 Ki > 10000 nM T15571 C6AV9G 145978819 Ki > 10000 nM T15571 C87MSW 145980271 Ki = 4152 nM T15571 CNJH37 145986752 Ki = 4973 nM T15571 CC2G1V 146025727 Ki = 6200 nM T15571 CV9G7Z 153287572 Ki > 10000 nM T15571 CO85KL 153287574 Ki > 10000 nM T15571 CB79ZW 155536080 Ki = 1995.26 nM T15571 C0OK3E 155551348 Ki = 8690 nM T15571 C3N9VU 10251906 Ki > 500 nM T15571 CP9TR0 10324985 Ki = 228.6 nM T15571 CQ1LV7 135508617 Ki = 6725 nM T15571 D00CRA 1574 Ki > 10000 nM T15571 D00GSD 25107716 Ki = 178 nM T15571 D00OBS 44559159 Ki > 10000 nM T15571 D00VRV 10171 Ki < 10 nM T15571 D01HRV 9847194 IC50 > 10000 nM T15571 D01KAX 135453290 Ki > 10000 nM T15571 D01WWC 16573 Ki = 566 nM T15571 D02UWB 1809 Ki = 20 nM T15571 D03DET 10287730 Ki = 3162.28 nM T15571 D03LPH 107838 Ki = 3200 nM T15571 D03TDN 1342 Ki = 40 nM T15571 D03XKU 44455986 Ki = 24 nM T15571 D03ZHB 44455973 Ki = 84.4 nM T15571 D04TPO 16006492 Ki = 5.012 nM T15571 D04UTQ 12683497 Ki = 2800 nM T15571 D05EQG 5265 Ki = 63000 nM T15571 D05GDP 599482 Ki > 10000 nM T15571 D07XTU 1229 Ki > 1000 nM T15571 D08OFG 11177588 Ki > 10000 nM T15571 D08VGJ 9904281 Ki = 43 nM T15571 D09HJL 10331436 Ki > 10000 nM T15571 D09RPR 16737207 Ki > 10000 nM T15571 D09WIL 10028436 Ki = 168 nM T15571 D0C3AR 44456244 Ki = 892 nM T15571 D0C5GF 6918515 Ki = 5160 nM T15571 D0CK9K 6918513 Ki = 4620 nM T15571 D0D1PE 169339 Ki > 10000 nM T15571 D0EA7Z 44455983 Ki = 805 nM T15571 D0F6CD 5202 Ki = 82 nM T15571 D0FF6S 16038374 IC50 > 10000 nM T15571 D0I6II 45263885 Ki = 658 nM T15571 D0J2UA 135433933 Ki = 9621 nM T15571 D0L5MW 181743 Ki = 2224 nM T15571 D0M2ZE 6604756 Ki = 168 nM T15571 D0O3GF 1220 Ki = 1000 nM T15571 D0W2YN 2760172 Ki = 2100 nM T15571 D0X1QW 122334 Ki = 2331 nM T15571 D0X6MT 4106 Ki = 1 nM T15571 D0X9YS 23642275 Ki = 98.5 nM T15571 D0XX2U 16006606 Ki = 6.3 nM T15571 D0Y9TL 13702393 Ki = 99 nM T12241 D08HZC 5852 IC50 = 270000 nM T12241 CVQR28 168091 IC50 = 40000 nM T12241 CE7M6K 269624 IC50 = 6300 nM T12241 CKFD03 439742 IC50 = 14000 nM T12241 C89ZER 2746654 IC50 = 6000 nM T12241 C8O4KD 5281599 IC50 > 400000 nM T12241 C3ZJ8U 5281609 IC50 > 400000 nM T12241 CDBE15 5947235 IC50 > 100000 nM T12241 CGH12F 6436272 IC50 = 1100 nM T12241 CU6W4G 6789060 IC50 = 6000 nM T12241 CX8V7B 6832311 IC50 = 5000 nM T12241 C1JGO8 9557956 IC50 = 40000 nM T12241 CSJ73Q 10347674 IC50 > 400000 nM T12241 CG56QX 13128573 IC50 = 50000 nM T12241 CS56LP 49822436 IC50 > 400000 nM T12241 CX1Y4Q 135517155 IC50 > 100000 nM T12241 CYCK69 145950009 IC50 > 100000 nM T12241 CY0CA3 145950025 IC50 = 2000 nM T12241 CBJE91 145950525 IC50 = 15000 nM T12241 CQ7TR0 145950586 IC50 = 6000 nM T12241 C7HIR2 145950806 IC50 = 15000 nM T12241 C09VKF 145951046 IC50 = 6000 nM T12241 CMD12Q 145951265 IC50 > 100000 nM T12241 CN8O3L 145951907 IC50 = 30000 nM T12241 CE0LR1 145952322 IC50 = 12000 nM T12241 CG5IR7 145952829 IC50 = 3000 nM T12241 CFYH93 145952906 IC50 = 12000 nM T12241 CID02M 145953955 IC50 = 3500 nM T12241 CYA18C 145954124 IC50 = 2100 nM T12241 CID9L8 145954253 IC50 = 40000 nM T12241 C9EV7T 145954518 IC50 > 100000 nM T12241 CU0N7F 145954660 IC50 = 6000 nM T12241 CWT0C2 145954999 IC50 = 10000 nM T12241 C4A7EB 145955194 IC50 = 2000 nM T12241 CC34VO 145955249 IC50 = 2500 nM T12241 CV6JN2 145955896 IC50 = 2700 nM T12241 CU0I6G 145956477 IC50 > 100000 nM T12241 CQN7K8 145956633 IC50 = 1900 nM T12241 CY5OA8 145957277 IC50 = 7000 nM T12241 CVJ8Q7 145957412 IC50 = 2000 nM T12241 C21RHB 145957746 IC50 = 2000 nM T12241 CP74VC 145958243 IC50 = 25000 nM T12241 C2Q9PB 145958460 IC50 = 10000 nM T12241 CD0L9T 145958807 IC50 > 400000 nM T12241 C8AK7F 145959104 IC50 = 6000 nM T12241 C7EX3J 145959358 IC50 = 15000 nM T12241 COW3Z4 145959534 IC50 = 1200 nM T12241 C8PQC2 145959639 IC50 > 100000 nM T12241 CDQ90E 145959869 IC50 = 6000 nM T12241 C1WQP3 145971246 IC50 = 3000 nM T12241 CU61TX 145972452 IC50 = 6000 nM T12241 CK05FS 145974829 IC50 = 5000 nM T12241 D01BTV 286 IC50 = 570 nM T57278 D03ZBT 11626560 IC50 > 1000 nM T57278 D09KTS 24821094 IC50 > 1000 nM T57278 D0E6XR 3062316 IC50 = 137 nM T57278 D03HUX 49792852 IC50 > 10000 nM T57278 D04AHQ 71721540 IC50 = 20 nM T57278 D04SLF 9903 IC50 = 50000 nM T57278 D0E3TC 44259 IC50 = 74.5 nM T57278 D03BNU 59604787 IC50 > 10000 nM T57278 D0T3ME 156422 IC50 = 160 nM T57278 CT52XN 92997 IC50 = 39810.72 nM T57278 CXQ5O3 115245 IC50 = 48977.88 nM T57278 CY13FW 644243 IC50 = 760 nM T57278 C4RUV5 5329453 IC50 = 250 nM T57278 C5GE7T 9917045 IC50 = 5200 nM T57278 CSGD16 10246246 IC50 > 7000 nM T57278 CBOP58 11293798 Ki > 10000 nM T57278 C26BZX 11362471 Ki > 10000 nM T57278 CWXB93 11397177 Ki > 10000 nM T57278 C35EIU 11698847 IC50 > 316227.77 nM T57278 C45EWD 11723489 IC50 > 7000 nM T57278 CP7AH3 11755812 IC50 = 35 nM T57278 CFPW41 16007116 Ki > 8000 nM T57278 C6JV7W 23400934 IC50 > 7000 nM T57278 CD5S7O 23401001 IC50 > 7000 nM T57278 CA3I4T 24753787 IC50 > 50000 nM T57278 CY8L7E 24896769 IC50 > 10000 nM T57278 C6W5LZ 25081574 IC50 = 4100 nM T57278 CA98KR 44432441 IC50 > 10000 nM T57278 C3VRO9 44557921 IC50 > 10000 nM T57278 C3HW7L 44570553 IC50 > 30000 nM T57278 C17PVE 44570554 IC50 > 30000 nM T57278 CLOY92 44570599 IC50 = 3000 nM T57278 CK06LT 44570600 IC50 > 30000 nM T57278 CY3HW5 46224684 IC50 > 10000 nM T57278 CYT37A 46232443 IC50 > 50000 nM T57278 C48ZVW 46232555 IC50 = 4400 nM T57278 CS9B1U 46232556 IC50 = 5200 nM T57278 CLS29B 46872626 IC50 > 10000 nM T57278 C2O8RZ 46886323 IC50 = 370 nM T57278 C0WYM1 46898022 IC50 = 10000 nM T57278 CF91RS 49843531 IC50 > 10000 nM T57278 CQ3KU9 50899556 IC50 = 260 nM T57278 C2Y6QS 50938552 IC50 > 10000 nM T57278 C61DVY 50990961 IC50 = 18 nM T57278 CV3UP9 50992247 IC50 = 11 nM T57278 CS9G6E 50997096 IC50 > 10000 nM T57278 C9NYP4 51036677 IC50 > 10000 nM T57278 C4WRY3 51037112 IC50 > 10000 nM T57278 CRI28Z 51037948 IC50 > 10000 nM T57278 C3LB5V 52941849 IC50 > 10000 nM T57278 CW2X5E 52944268 IC50 = 740 nM T57278 C9PX2J 52945752 IC50 = 300 nM T57278 CL4ED3 52945753 IC50 = 840 nM T57278 CIR3Q0 52947964 IC50 = 5600 nM T57278 C09SDH 53257410 IC50 > 10000 nM T57278 CBK9Q6 53357848 IC50 > 10000 nM T57278 C8NA4L 53384644 IC50 = 16000 nM T57278 CPHX64 57325478 IC50 > 50000 nM T57278 CQ9BW4 57325479 IC50 > 50000 nM T57278 CVK0G4 58056356 IC50 > 50000 nM T57278 CT3EW2 59292007 IC50 > 1000 nM T57278 C9ZCT2 62705065 IC50 > 1000 nM T57278 C10AMI 66553589 IC50 = 6180 nM T57278 CV63UL 67240318 IC50 > 10000 nM T57278 C23UCM 70946730 IC50 = 300 nM T57278 CKT60L 71455860 Ki > 2800 nM T57278 CCN01X 71547862 IC50 > 10000 nM T57278 CVIA91 71553085 IC50 = 30000 nM T57278 C1TR3O 71553152 IC50 = 30000 nM T57278 CF8Z9P 71604568 IC50 = 19952.62 nM T57278 CP5T7A 71604569 IC50 = 30902.95 nM T57278 CG6SI4 71604570 IC50 = 23988.33 nM T57278 CD1PS3 71604720 IC50 = 17378.01 nM T57278 CN3FH0 71604721 IC50 = 101000 nM T57278 C13PNG 71604722 IC50 = 60255.96 nM T57278 CB8KL7 71604723 IC50 > 316227.77 nM T57278 C01POC 71604724 IC50 > 316227.77 nM T57278 C24DHJ 71604873 IC50 > 316227.77 nM T57278 CR4D9H 71604874 IC50 = 26000 nM T57278 CUGT42 71604875 IC50 = 27542.29 nM T57278 CJDA65 71604876 IC50 = 6606.93 nM T57278 CEK72C 71604877 IC50 = 7585.78 nM T57278 CW6NK4 71605036 IC50 = 50118.72 nM T57278 CX3E8O 71605037 IC50 = 100000 nM T57278 C60QZJ 71605038 IC50 = 20417.38 nM T57278 CZHF09 71716449 IC50 >= 100000 nM T57278 C7H6GC 71717050 IC50 = 6300 nM T57278 CV2HP0 71717673 IC50 >= 100000 nM T57278 CN56HF 71718279 IC50 >= 100000 nM T57278 C9E3XT 71718280 IC50 = 14000 nM T57278 CQL9G2 71718885 IC50 = 24000 nM T57278 CSEQ21 71719490 IC50 > 100000 nM T57278 CQ36JS 71719491 IC50 = 13000 nM T57278 CN6CA9 71720086 IC50 = 94000 nM T57278 C46ONG 71720087 IC50 = 29000 nM T57278 C4TRW2 71720468 IC50 > 316227.77 nM T57278 CR97JV 71720738 IC50 = 71000 nM T57278 CBX0N9 71720739 IC50 = 15000 nM T57278 C60TUV 72737208 IC50 > 10000 nM T57278 CJ3WA6 72737404 IC50 > 10000 nM T57278 CVNW01 73386831 IC50 > 1000 nM T57278 CCJ43A 86302281 IC50 > 10000 nM T57278 CB5NJ4 86302541 IC50 > 10000 nM T57278 CPG3A5 86302574 IC50 > 30000 nM T57278 CY0UC4 90645194 IC50 > 10000 nM T57278 CX29IY 90655145 IC50 > 10000 nM T57278 CAPB10 91666638 IC50 = 160 nM T57278 CY7BI2 118706214 IC50 > 10000 nM T57278 CKM13G 118710440 IC50 = 1190 nM T57278 CVJ7A8 118710441 IC50 = 1470 nM T57278 CSRQ30 118710442 IC50 = 2500 nM T57278 C4E0UV 118710443 IC50 = 750 nM T57278 CA1ZY6 118710444 IC50 = 2310 nM T57278 COJ3U8 118710445 IC50 = 680 nM T57278 CDTF80 118710446 IC50 = 580 nM T57278 C0D1PA 118710447 IC50 = 730 nM T57278 C6BH8K 118710448 IC50 = 720 nM T57278 CDLQ85 118710449 IC50 = 620 nM T57278 C9M5ZO 118710451 IC50 = 960 nM T57278 C28ABH 118710452 IC50 = 3210 nM T57278 CO8C6F 118710453 IC50 = 200 nM T57278 CR4S3Y 118710454 IC50 = 170 nM T57278 C7E0VG 118710455 IC50 = 450 nM T57278 C78JUP 118710456 IC50 = 230 nM T57278 CC70YB 118710457 IC50 = 320 nM T57278 CQCX41 118737057 IC50 = 16 nM T57278 C8KXV1 127025843 IC50 > 1000 nM T57278 C40DLR 127035199 IC50 = 4265.8 nM T57278 CN3F9G 127035350 IC50 = 89125.09 nM T57278 C0OM1N 127035351 IC50 = 6309.57 nM T57278 CEV2H1 127035714 IC50 = 8912.51 nM T57278 CO7SQ1 127035899 IC50 > 100000 nM T57278 C9WGB8 127035904 Ki = 1400 nM T57278 CCLF46 127035905 IC50 > 100000 nM T57278 C06KQV 127035906 IC50 = 22387.21 nM T57278 CVU98P 127035907 Ki = 2400 nM T57278 CDI68C 127035908 IC50 = 47863.01 nM T57278 C6TJF3 127036098 IC50 > 100000 nM T57278 CD98XV 127036099 IC50 = 50118.72 nM T57278 CFSP72 127036100 IC50 = 5011.87 nM T57278 CKIA98 127036101 IC50 = 4073.8 nM T57278 CKX40V 127037812 IC50 > 10000 nM T57278 C70RUP 127038480 IC50 > 10000 nM T57278 C3WCN8 127041777 IC50 > 10000 nM T57278 CHK16Q 127045929 IC50 > 1000 nM T57278 CY3J0C 127047591 IC50 > 1000 nM T57278 CERS64 132937256 IC50 > 30000 nM T57278 CN35SO 134146628 IC50 > 1000 nM T57278 CYL5V1 134694986 IC50 > 30000 nM T57278 CDT7E4 136211077 IC50 > 100 nM T57278 CXC69T 137321158 IC50 = 341 nM T57278 C25ERN 137631967 IC50 > 100 nM T57278 C06JRX 137637094 IC50 > 10 nM T57278 CTD9I4 137637448 Ki > 15000 nM T57278 C1DK0P 137651391 IC50 > 100 nM T57278 CSB0L1 137654726 IC50 = 5000 nM T57278 CV5H3Z 137657932 IC50 > 10 nM T57278 CSRI06 138547901 IC50 > 1000 nM T57278 CUXO19 138617501 IC50 > 1000 nM T57278 CO9P7G 145351804 IC50 > 1000 nM T57278 C29XUO 145945978 IC50 > 1000 nM T57278 C4OD9Q 145967187 IC50 > 1000 nM T57278 CUJS82 145969463 IC50 = 4900 nM T57278 COD32L 145970693 IC50 = 4100 nM T57278 C2MD1Q 155513187 IC50 > 10000 nM T57278 CS69CA 155532132 IC50 = 13.5 nM T57278 D00ERW 44444843 Ki > 8000 nM T57278 D02BXJ 46864270 IC50 = 0.6 nM T57278 D05FXD 44478401 IC50 = 2.3 nM T57278 D0C2GE 67161540 IC50 = 1700 nM T57278 D0O6OH 71553154 IC50 = 2430 nM T57278 D0X8BU 71718651 IC50 = 2041.74 nM T57278 D0Y0BK 11524144 IC50 = 11 nM T01385 D09GOS 2812 IC50 = 1400 nM T01385 D08OOJ 73051434 IC50 = 11 nM T01385 D0F6NT 1162727 IC50 > 30000 nM T01385 C05ZPG 397069 IC50 > 100000 nM T01385 C86FWD 470278 IC50 > 100000 nM T01385 C5EY0V 672872 IC50 = 80 nM T01385 CHXJ51 697280 IC50 = 190 nM T01385 CR98CN 704363 IC50 = 230 nM T01385 C1IV9D 704494 IC50 = 290 nM T01385 C4X1BC 704553 IC50 = 300 nM T01385 CYF9E1 720920 IC50 > 30000 nM T01385 C1QRW7 768027 IC50 = 2000 nM T01385 C30HYZ 788482 IC50 = 1290 nM T01385 C34XJV 793670 EC50 = 90 nM T01385 C9M6JL 863286 IC50 > 30000 nM T01385 C1KQL0 864171 IC50 > 30000 nM T01385 C8KUR0 865869 IC50 = 9920 nM T01385 C3FX5T 865870 IC50 = 2690 nM T01385 C7MLU1 877530 IC50 > 10000 nM T01385 CHX2D5 877815 IC50 = 430 nM T01385 CA0J3M 906598 IC50 > 100000 nM T01385 CD7O0J 935549 IC50 = 4800 nM T01385 CPL20I 973124 IC50 = 1300 nM T01385 CZ32JI 2249447 IC50 = 8300 nM T01385 C5Q0HK 2975404 IC50 > 37000 nM T01385 CX3JD7 3556408 IC50 = 760 nM T01385 CEM5C8 25100438 IC50 = 360 nM T01385 C07VAB 25100440 IC50 = 670 nM T01385 CDXT96 30869108 IC50 = 990 nM T01385 C1M5SP 45019715 IC50 > 30000 nM T01385 CH2V5M 46865782 IC50 = 120 nM T01385 C9P6UC 46880290 IC50 > 20000 nM T01385 CGIA46 46880328 IC50 = 2700 nM T01385 C3VKZ8 46880369 IC50 = 180 nM T01385 CZHM28 46880414 IC50 = 91 nM T01385 CAU6O0 46880464 IC50 = 120 nM T01385 CXDK90 46880466 IC50 = 140 nM T01385 CVEC92 46880467 IC50 = 170 nM T01385 CHW21A 46880468 IC50 = 190 nM T01385 C2YWI1 46880469 IC50 = 330 nM T01385 CBQ49H 46880502 IC50 = 130 nM T01385 CA6IV3 46880503 IC50 = 230 nM T01385 CZPV27 49830258 IC50 = 110 nM T01385 C7EY1H 49852176 IC50 > 5000 nM T01385 C4VIP1 50918580 IC50 = 425 nM T01385 C9OJG1 52374396 IC50 > 30000 nM T01385 CCR7O0 54670937 IC50 > 5000 nM T01385 CM59RJ 56928016 IC50 > 5000 nM T01385 CH65ZE 57328756 IC50 = 22000 nM T01385 C1XBG6 58523937 IC50 > 5000 nM T01385 C07XGU 71520305 IC50 = 88 nM T01385 CWZ27A 71520306 IC50 = 90 nM T01385 C5WQ8Z 71520307 IC50 = 100 nM T01385 CN4O3X 71520308 IC50 = 134 nM T01385 C5OK4Z 71520309 IC50 = 150 nM T01385 C6SRU5 71520310 IC50 = 184 nM T01385 C82ATI 71520425 IC50 = 225 nM T01385 C2B9KN 71520426 IC50 = 257 nM T01385 CQ1JY3 71520427 IC50 = 443 nM T01385 CZ80NI 71520429 IC50 = 43 nM T01385 CB4JG8 71520430 IC50 = 48 nM T01385 C13YPQ 71520540 IC50 = 71 nM T01385 CO2QT1 71520541 IC50 = 41 nM T01385 CI8B7L 71520542 IC50 = 42 nM T01385 CKQL06 71520543 IC50 = 63 nM T01385 CY6PL1 71520544 IC50 = 65 nM T01385 CE4Q0T 71520634 IC50 = 112 nM T01385 CMQ68E 71520635 IC50 = 162 nM T01385 CP9UY2 71520818 IC50 > 30000 nM T01385 C7HFN3 71520819 IC50 = 960 nM T01385 CS90CX 71520820 IC50 = 720 nM T01385 CPB6S5 71520821 IC50 = 960 nM T01385 C4K1AN 71520822 IC50 = 1150 nM T01385 C45XQJ 71520919 IC50 > 30000 nM T01385 C7V2LX 71520920 IC50 = 3790 nM T01385 C0F5TW 71520926 IC50 = 172 nM T01385 CBO1H8 71520927 IC50 = 262 nM T01385 C1BSM0 71520928 IC50 = 523 nM T01385 CR42SU 71520929 IC50 = 683 nM T01385 C6I0OW 71520930 IC50 = 976 nM T01385 COYE37 71520931 IC50 = 1236 nM T01385 CEHQ96 71521025 IC50 > 30000 nM T01385 C4KCX9 71521026 IC50 > 30000 nM T01385 CEYG08 71521027 IC50 > 30000 nM T01385 CU10JB 71521028 IC50 = 2250 nM T01385 C1YF8L 71521029 IC50 = 1960 nM T01385 CIG40P 71521030 IC50 = 19430 nM T01385 C5IH4G 71521031 IC50 > 30000 nM T01385 CT4O1M 71521032 IC50 = 2031 nM T01385 CH97TQ 71521033 IC50 = 536 nM T01385 CXG73H 71521034 IC50 = 379 nM T01385 CZMO73 71521035 IC50 = 1394 nM T01385 C8F3AT 71521036 IC50 = 451 nM T01385 C9YN6X 71521037 IC50 = 908 nM T01385 C27VGT 71521131 IC50 = 1880 nM T01385 CT7IQ3 71521132 IC50 = 2060 nM T01385 C1N0IP 71521133 IC50 = 2320 nM T01385 C9EJZ4 71521134 IC50 = 16220 nM T01385 C8AR7M 71521135 IC50 > 30000 nM T01385 CG1XD3 71521136 IC50 = 19600 nM T01385 C3H7PS 71521137 IC50 > 30000 nM T01385 C6X8OQ 71521138 IC50 = 71 nM T01385 C10NRW 71521139 IC50 = 58 nM T01385 C7H1ME 71521140 IC50 = 25 nM T01385 CK6M1Y 71521141 IC50 = 54 nM T01385 CI0DC4 71521236 IC50 = 2690 nM T01385 C4R3FX 71521237 IC50 = 740 nM T01385 C3AJ2W 71521238 IC50 = 960 nM T01385 CS5E0K 71521239 IC50 = 2780 nM T01385 CVSF75 71521240 IC50 = 53 nM T01385 CIY79B 71521241 IC50 = 67 nM T01385 C0K3FZ 71521347 IC50 = 2810 nM T01385 CDR29I 71521348 IC50 > 30000 nM T01385 C4P1OI 71521349 IC50 > 30000 nM T01385 C2FU7P 71521350 IC50 > 30000 nM T01385 CSP46C 71521351 IC50 > 30000 nM T01385 C2F8TA 71521352 IC50 = 470 nM T01385 CVYJ16 71521353 IC50 > 30000 nM T01385 CR1LF6 71521458 IC50 = 1290 nM T01385 CDF30Z 71521459 IC50 = 2400 nM T01385 CU9D2H 71521460 IC50 = 7730 nM T01385 C2H9UV 71521461 IC50 = 11780 nM T01385 CG8Z3S 71521462 IC50 = 26720 nM T01385 C7CF8N 71521463 IC50 > 30000 nM T01385 CM7UB5 71521536 IC50 = 440 nM T01385 C46IZM 71521537 IC50 = 18640 nM T01385 C21MUO 71521538 IC50 = 2860 nM T01385 CS43JP 71521539 IC50 = 1940 nM T01385 CMUZ53 71521540 IC50 = 8720 nM T01385 CE1FJ6 71521541 IC50 = 11170 nM T01385 CQ0BK1 71521542 IC50 > 30000 nM T01385 CBJM79 71521620 IC50 > 30000 nM T01385 CY8RF0 71521621 IC50 = 1970 nM T01385 CV4Q5F 71521622 IC50 = 4300 nM T01385 CJ9B0Z 71521623 IC50 > 30000 nM T01385 CS84PN 71521624 IC50 = 2850 nM T01385 CX6Z8C 71521625 IC50 = 3450 nM T01385 CTK92X 71521626 IC50 = 5560 nM T01385 CPF75N 71521709 IC50 = 1277 nM T01385 CPJ3Q1 71521710 IC50 = 279 nM T01385 CP82UW 71521711 IC50 = 283 nM T01385 CXRZ18 71521712 IC50 = 379 nM T01385 C3W9KG 71521713 IC50 = 524 nM T01385 CN96LY 71521714 IC50 = 3129 nM T01385 CLD68Y 71521715 IC50 = 375 nM T01385 C5WV4I 71521791 IC50 = 140 nM T01385 C93NYA 71521792 IC50 = 168 nM T01385 CSH67K 71521793 IC50 = 604 nM T01385 C7KRB8 71521794 IC50 = 220 nM T01385 C7IU9X 71521795 IC50 = 609 nM T01385 C23LYC 71521796 IC50 = 587 nM T01385 CRO46G 71521797 IC50 = 71 nM T01385 CH1KQ4 71604308 IC50 = 760 nM T01385 CEA94U 71604309 IC50 = 1100 nM T01385 CC1V2S 71607189 IC50 = 370 nM T01385 C4TG6V 72721010 IC50 = 43 nM T01385 C2R9LK 73051132 IC50 = 445 nM T01385 C1M0KD 73051133 IC50 = 153 nM T01385 CG71JS 73051280 IC50 = 47 nM T01385 C1NQ8H 73051924 IC50 = 98 nM T01385 C7IMZ0 73052240 IC50 = 3134 nM T01385 C4HM1G 73052241 IC50 = 76 nM T01385 C4FWO9 73052243 IC50 > 5000 nM T01385 C3VLG0 73052401 IC50 = 95 nM T01385 C79HDC 73052716 IC50 = 1790 nM T01385 CEG8R1 73052718 IC50 = 192 nM T01385 CTR3G9 73052878 IC50 = 6 nM T01385 C0VA6M 73053029 IC50 = 304 nM T01385 C95DXT 82192375 IC50 > 37000 nM T01385 C46GEV 89927846 IC50 = 370 nM T01385 C9W7GE 89927907 IC50 = 3000 nM T01385 CBC03Z 89927958 IC50 = 152 nM T01385 CRX36D 89927984 IC50 = 145 nM T01385 CC36BE 89928011 IC50 = 233 nM T01385 C0XAP3 89928021 IC50 = 248 nM T01385 CMI21Z 89928023 IC50 = 68 nM T01385 CYEC61 89928082 IC50 > 5000 nM T01385 C0J7BI 89928094 IC50 = 149 nM T01385 CE81KH 89928101 IC50 = 144 nM T01385 CTGD01 89928106 IC50 = 2075 nM T01385 C6WS8V 89928107 IC50 = 632 nM T01385 CK7GM3 89928109 IC50 = 795 nM T01385 CDP70Y 89928159 IC50 = 227 nM T01385 C29ART 89928200 IC50 = 342 nM T01385 C7PH3D 89928222 IC50 = 180 nM T01385 C8AZT1 89928224 IC50 = 1068 nM T01385 CBK1W6 89941289 IC50 > 5000 nM T01385 CB8IQ2 90031714 IC50 > 5000 nM T01385 CN91SG 90032051 IC50 = 651 nM T01385 CJZS64 90032070 IC50 = 367 nM T01385 CY5TU6 90032147 IC50 = 3912 nM T01385 C9ISK1 90032171 IC50 = 215 nM T01385 CNE9B5 90032547 IC50 = 8908 nM T01385 C2XC7V 90032634 IC50 = 648 nM T01385 CBTL19 101907906 IC50 = 26300 nM T01385 CA6E9Y 101910775 IC50 = 61 nM T01385 CMY30U 101910777 IC50 = 74 nM T01385 C1A8JZ 114286471 IC50 = 70 nM T01385 CMA84J 117094775 IC50 = 907 nM T01385 CF2RD3 118322226 IC50 = 4832 nM T01385 CQBG03 118724369 IC50 = 21600 nM T01385 CD71XN 118724370 IC50 = 20500 nM T01385 CEC71H 118724371 IC50 > 37000 nM T01385 CF53BA 118724372 IC50 > 37000 nM T01385 C5RFT0 118724373 IC50 = 15400 nM T01385 CH8PF1 118724374 IC50 > 37000 nM T01385 C9C4WZ 118724375 IC50 = 2600 nM T01385 C9SLR5 118724376 IC50 = 8700 nM T01385 CYX0K4 118724377 IC50 > 37000 nM T01385 COE61I 118724378 IC50 > 37000 nM T01385 CS8YZ3 118724379 IC50 = 11400 nM T01385 C9RJV7 118724380 IC50 = 4800 nM T01385 CA3LT6 118724381 IC50 > 37000 nM T01385 CE43MW 118724382 IC50 = 2700 nM T01385 CH42TP 118724383 IC50 = 2600 nM T01385 CQFZ65 118724384 IC50 = 8400 nM T01385 CYV7T4 118724385 IC50 > 37000 nM T01385 C2SV1M 118724386 IC50 = 300 nM T01385 CYLT37 118724387 IC50 = 673 nM T01385 CA93NZ 118724388 IC50 = 141 nM T01385 CV56WG 118724389 IC50 = 700 nM T01385 C7LCP1 118724390 IC50 = 3041 nM T01385 C7XV4F 118724391 IC50 = 578 nM T01385 CD2WN1 118724392 IC50 = 552 nM T01385 C9FVI6 118724393 IC50 = 483 nM T01385 C0O3AC 118724394 IC50 = 543 nM T01385 C82IQE 118724395 IC50 = 116 nM T01385 CO9R3I 118724396 IC50 = 201 nM T01385 CRF7Z9 118724397 IC50 = 879 nM T01385 C5N1SJ 118724762 IC50 = 577 nM T01385 CG01LE 118724763 IC50 = 742 nM T01385 CA39KG 118724764 IC50 = 221 nM T01385 C1JTS3 118724765 IC50 = 921 nM T01385 CK7Y9N 118724766 IC50 = 1091 nM T01385 CCM3X6 118724767 IC50 = 2189 nM T01385 CAMZ23 118724768 IC50 = 112 nM T01385 CHZ6K1 118724769 IC50 = 60 nM T01385 C5T1RV 118724770 IC50 = 150 nM T01385 CZKE26 118724771 IC50 = 570 nM T01385 CGP36N 118724772 IC50 = 1201 nM T01385 C3YPM4 118724773 IC50 = 1667 nM T01385 C3K2BJ 118724774 IC50 = 2188 nM T01385 CYJR42 118724775 IC50 = 27 nM T01385 CF5X3Y 118724776 IC50 = 36 nM T01385 C7UZ5H 118724777 IC50 = 4313 nM T01385 CO6GN4 118724778 IC50 > 10000 nM T01385 CPK72W 118724779 IC50 = 127 nM T01385 CGO35H 118724780 IC50 = 448 nM T01385 C96YAG 118724781 IC50 = 133 nM T01385 CJ1UK5 118724782 IC50 = 264 nM T01385 C8DX9G 118724783 IC50 = 986 nM T01385 CN49SF 118724784 IC50 = 9288 nM T01385 CA78KC 118724785 IC50 = 1691 nM T01385 CL25HP 118724786 IC50 = 6939 nM T01385 CEG6T2 118724787 IC50 = 7108 nM T01385 C32LRP 118724788 IC50 = 8860 nM T01385 C43QNY 118724789 IC50 = 1679 nM T01385 CCDH40 118724790 IC50 = 474 nM T01385 CA6F9K 118724791 IC50 = 2762 nM T01385 CV5P0J 118724792 IC50 = 5645 nM T01385 CWQ61D 118724793 IC50 = 4608 nM T01385 CKM04D 118724794 IC50 = 7610 nM T01385 CTRV82 118724795 IC50 = 2181 nM T01385 C69HKQ 118724796 IC50 = 2433 nM T01385 CO9W1I 118724797 IC50 = 3473 nM T01385 CLVO02 118724798 IC50 = 5036 nM T01385 CACB18 118724799 IC50 = 5165 nM T01385 C8LJ1X 118724800 IC50 > 10000 nM T01385 CCK45Q 118724801 IC50 = 46 nM T01385 C6B1FX 118724802 IC50 = 87 nM T01385 CY50JH 118724803 IC50 = 106 nM T01385 CS8O9F 118724804 IC50 = 135 nM T01385 C4SU7T 118724805 IC50 = 149 nM T01385 CW9E3Z 118724806 IC50 = 183 nM T01385 CY6C3R 118724807 IC50 = 237 nM T01385 C6H9CJ 118724808 IC50 = 59 nM T01385 CX7FM5 118724809 IC50 = 89 nM T01385 CE54NW 118724810 IC50 = 102 nM T01385 CXJ43Z 118724811 IC50 = 106 nM T01385 CVKT57 118724812 IC50 = 222 nM T01385 CZV40N 118724813 IC50 = 246 nM T01385 C4YH3Q 118724814 IC50 = 299 nM T01385 C0F8VX 118724815 IC50 = 82 nM T01385 C6QRS2 118724816 IC50 = 109 nM T01385 C3NK9E 118724817 IC50 = 452 nM T01385 C2DSR3 118724818 IC50 = 491 nM T01385 C4UJ7V 127031857 IC50 = 50 nM T01385 CT0F5Y 127032127 IC50 = 710 nM T01385 C3VG0W 127032128 IC50 = 3800 nM T01385 CGU32Y 127032429 IC50 = 4700 nM T01385 CVXR24 127032715 IC50 = 21500 nM T01385 CRN4B7 127032716 IC50 = 240 nM T01385 CKGU65 127039986 IC50 > 5000 nM T01385 CRB4C1 127039987 IC50 > 5000 nM T01385 C2GX8Z 127039988 IC50 > 5000 nM T01385 CV81YZ 127039989 IC50 = 3860 nM T01385 C6OQ4W 127039990 IC50 > 5000 nM T01385 CB2AR3 127040617 IC50 > 5000 nM T01385 CJ4FQ3 127040618 IC50 > 5000 nM T01385 CX0P2U 127040619 IC50 > 5000 nM T01385 C82QOL 127040620 IC50 > 5000 nM T01385 CWC4M7 127040621 IC50 > 5000 nM T01385 CWA09O 127040622 IC50 > 5000 nM T01385 CQ6KV5 127041309 IC50 = 15 nM T01385 CI0X6E 127041536 IC50 > 5000 nM T01385 CQ2VO1 127041608 IC50 = 71 nM T01385 CGN9I7 127041609 IC50 = 23 nM T01385 C3TUR2 127041878 IC50 > 5000 nM T01385 CR8PG7 127041879 IC50 > 5000 nM T01385 CV92NA 129073433 IC50 = 180 nM T01385 C3IN1Q 132561319 IC50 = 7900 nM T01385 C1LN3T 132570328 IC50 = 160 nM T01385 C3H6DA 132570329 IC50 = 44 nM T01385 C6H9BZ 132570331 IC50 = 31400 nM T01385 CEZ9B2 139035043 IC50 = 7200 nM T01385 CEX63L 139298248 IC50 = 7 nM T01385 C10RBQ 140939034 IC50 = 90 nM T01385 CKW53D 140939044 IC50 = 100 nM T01385 C8CQT0 140939054 IC50 = 280 nM T01385 C7TX2S 140939070 IC50 = 190 nM T01385 COWD30 140939079 IC50 = 20 nM T01385 C4V7CI 140939088 IC50 = 2610 nM T01385 C2C9PG 140939100 IC50 = 1130 nM T01385 C6PN5R 140939111 IC50 = 200 nM T01385 C0ZH4R 140939116 IC50 = 800 nM T01385 CTJ0U5 140939119 IC50 = 19000 nM T01385 CGLY18 140939126 IC50 = 210 nM T01385 CUC3P9 140939138 IC50 = 1060 nM T01385 CW8U7Q 140939163 IC50 = 4760 nM T01385 CZ0XI5 140939170 IC50 = 1050 nM T01385 CX7F5D 140939178 IC50 = 50 nM T01385 CP7Q2G 140939185 IC50 = 330 nM T01385 C4JAX8 145988686 IC50 = 380 nM T01385 C7LGD3 154730745 Ki = 33.2 nM T01385 CDN0B5 155068296 IC50 = 82.8 nM T01385 C9YQ7I 155510447 Ki = 20.8 nM T01385 C43MSR 155510502 Ki = 28.1 nM T01385 CQV4H6 155513260 Ki = 32.8 nM T01385 C3K1VZ 155513650 IC50 = 119.7 nM T01385 CSB62H 155515179 Ki = 24.5 nM T01385 CN98ID 155517954 IC50 = 922.1 nM T01385 CD0A2C 155518618 Ki = 40.8 nM T01385 CM48LB 155522046 IC50 = 34.6 nM T01385 CR34KJ 155522981 Ki = 26.6 nM T01385 C0CA1Z 155524986 Ki = 43 nM T01385 CWTP12 155527743 Ki = 32.3 nM T01385 CZA90T 155528495 IC50 = 36.4 nM T01385 C0HU1L 155528572 IC50 = 134.9 nM T01385 CG8Z9A 155530177 Ki = 30.6 nM T01385 C69LKC 155530248 Ki = 37.3 nM T01385 CBQ3N1 155533126 IC50 = 192.6 nM T01385 C80XHD 155536273 IC50 = 387.1 nM T01385 CWZS75 155538655 IC50 = 8 nM T01385 C9KO2J 155545885 IC50 = 129.4 nM T01385 C3VHG0 155547513 Ki = 42.4 nM T01385 CYFP96 155547774 Ki = 24.1 nM T01385 CLV2Z5 155555002 Ki = 26.9 nM T01385 C42ONM 155556308 IC50 = 448.7 nM T01385 C1QNZ5 155557365 Ki = 18.6 nM T01385 CGYS98 155557471 Ki = 37.9 nM T01385 CL28DA 155561627 IC50 = 160.9 nM T01385 C2M7QB 155561797 IC50 = 447.2 nM T01385 C3FXR6 155563226 IC50 = 100.9 nM T01385 C4LU8S 155563972 IC50 = 5104.5 nM T01385 CPU5R9 155564364 IC50 = 308.1 nM T01385 CIYS74 155565460 Ki = 31.4 nM T01385 D00YNY 753704 EC50 < 1200 nM T01385 D0D8SU 71521142 IC50 = 24 nM T57818 D0RA5Q 72172 IC50 = 160000 nM T57818 CK8VJ3 5311145 Ki > 1000000 nM T57818 CP4VT2 13633258 Ki = 51 nM T57818 CT3L5Q 14542146 Ki = 130000 nM T57818 CP4OT8 14542149 Ki = 170 nM T57818 CE1P6J 15719279 Ki = 1500 nM T57818 CD28WR 15719282 Ki = 3200 nM T57818 CYR87Z 15719283 Ki = 6500 nM T57818 CMWK71 44276411 Ki = 11 nM T57818 CS75VD 44360285 Ki > 300000 nM T57818 CVS46P 54394267 IC50 = 3500 nM T57818 D02BLC 20384324 Ki = 0.9 nM T57818 D0A7GO 44309732 Ki = 39000 nM T84117 D01AZG 5073 Ki > 1000 nM T84117 D0G8NN 119570 Ki > 10000 nM T84117 D0H3HM 60795 Ki > 1000 nM T84117 D0H7KF 5002 Ki > 1000 nM T84117 D0V4QS 135398745 Ki > 1000 nM T84117 D0Z1RV 135398737 Ki = 1000 nM T84117 D0Z6UC 5358 IC50 = 5500 nM T84117 D0N1HW 5311200 Ki > 10000 nM T84117 D0X2XF 177336 Ki < 10000 nM T84117 D02ZSO 6426760 IC50 > 10000 nM T84117 D03YPJ 5163 Ki < 5011.87 nM T84117 D0M7LV 5761 Ki = 93 nM T84117 D0Q2JS 10436045 Ki = 6.31 nM T84117 D0YP7L 6604889 Ki < 6309.57 nM T84117 C5H9CN 9287 Ki = 1905.46 nM T84117 C6WDL7 49756 Ki = 1800 nM T84117 CTB26S 52899 Ki > 10000 nM T84117 CKP25M 121881 Ki < 10000 nM T84117 C2VLP8 752521 Ki > 10000 nM T84117 CS8KE2 3649661 Ki > 10000 nM T84117 C0QCK1 6918455 Ki < 10000 nM T84117 CW0ZE5 6918542 Ki = 4220 nM T84117 CD0Z4I 6918648 Ki = 2511.89 nM T84117 CYMP40 9851789 IC50 = 99 nM T84117 CJW1P5 9888494 Ki < 10000 nM T84117 C3J8GU 9892409 Ki < 1000 nM T84117 CUN81Q 9905249 Ki > 10000 nM T84117 CYWQ50 9906447 Ki > 10000 nM T84117 C78MDV 9913554 Ki = 1584.89 nM T84117 CWO45F 9935387 Ki = 1000 nM T84117 CYH3R7 9947817 Ki = 770 nM T84117 C3S7XA 10009042 IC50 = 392 nM T84117 CV7R9F 10020040 Ki > 10000 nM T84117 CK18LT 10020895 Ki = 660 nM T84117 C4Q2SH 10249573 Ki < 10000 nM T84117 CMRA02 10257042 Ki < 6309.57 nM T84117 CH31DX 10267394 Ki > 10000 nM T84117 CU89JD 10314060 Ki > 10000 nM T84117 C9IAV3 10346043 Ki > 10000 nM T84117 C4TPN1 10413595 Ki > 10000 nM T84117 CD7U5I 10433930 Ki > 10000 nM T84117 COV85C 10472143 Ki = 280 nM T84117 CHE80N 10573876 Ki < 2511.89 nM T84117 CO23YX 10597140 Ki < 10000 nM T84117 C8MHZ9 10835110 Ki = 2511.89 nM T84117 CNB39C 10947658 Ki = 200 nM T84117 CVE8T3 11121216 Ki = 140 nM T84117 C9ZT5F 11536299 Ki > 10000 nM T84117 CGX8F6 11596869 Ki > 5370000 nM T84117 CXLW54 11948707 Ki > 10000 nM T84117 C8JQL7 11957735 IC50 > 10000 nM T84117 CZ2IS9 16660294 Ki > 10000 nM T84117 C7T8JC 19958494 Ki > 10000 nM T84117 C6LI5E 19958507 Ki > 10000 nM T84117 C3T5HF 21509921 Ki = 4045 nM T84117 CBN84K 22065997 Ki > 10000 nM T84117 CDC91N 24839550 Ki = 380.19 nM T84117 C3HK0J 24865725 Ki = 2511.89 nM T84117 C0O6FX 24865727 Ki > 10000 nM T84117 CI53SE 24893978 Ki > 10000 nM T84117 CA58DL 41305446 Ki > 10000 nM T84117 CC2OD4 44278111 Ki > 10000 nM T84117 CRMA84 44278114 Ki > 10000 nM T84117 CF0Y4M 44278115 Ki > 10000 nM T84117 CPWJ26 44343212 Ki < 10000 nM T84117 CUXH48 44352308 Ki > 4830 nM T84117 C4B0OI 44397588 Ki < 10000 nM T84117 C5FP0R 44397589 Ki < 10000 nM T84117 CE3G8U 44397670 Ki < 10000 nM T84117 CZL97F 44455426 Ki > 10000 nM T84117 C12XGE 44456400 Ki > 10000 nM T84117 C5ZML8 44457907 IC50 > 1000 nM T84117 CM3IR1 44457909 IC50 > 1000 nM T84117 CAS01K 44458044 IC50 > 1000 nM T84117 CGD04W 44458045 IC50 > 1000 nM T84117 C94DNM 44458229 IC50 > 1000 nM T84117 CM9YD2 44458486 IC50 > 1000 nM T84117 CRCH48 44582675 Ki > 10000 nM T84117 CEJ4R8 44582676 Ki > 10000 nM T84117 CZGP86 44582677 Ki > 10000 nM T84117 C5QB4K 44582678 Ki > 10000 nM T84117 C01RCI 44582705 Ki > 10000 nM T84117 CXL25V 44582706 Ki > 10000 nM T84117 C8MR1X 44582707 Ki > 10000 nM T84117 C4IT1N 44582708 Ki > 10000 nM T84117 C5ZDY3 46915370 Ki = 2900 nM T84117 C2LZJ0 49783209 Ki = 10000 nM T84117 C57SMG 49783415 Ki > 10000 nM T84117 C0TG6I 49783419 Ki > 10000 nM T84117 C2RY0J 50878551 Ki = 413 nM T84117 C1W6TV 50898777 Ki > 10000 nM T84117 CXMZ73 50898778 Ki > 10000 nM T84117 CE4KP1 51050257 Ki > 10000 nM T84117 C1TC7Q 56963799 Ki > 10000 nM T84117 C1LEH8 67268994 Ki = 1366 nM T84117 C3XNC2 71450247 Ki > 10000 nM T84117 CAQF34 71455625 Ki > 10000 nM T84117 CMJ1O9 71457409 Ki > 10000 nM T84117 C63YLA 71461049 Ki > 10000 nM T84117 CJD96I 71461050 Ki > 10000 nM T84117 C4P3JU 71462776 Ki > 10000 nM T84117 C3GUQ2 71462777 Ki > 10000 nM T84117 CC6Q5R 72771081 Ki < 100 nM T84117 CC65OA 73213195 Ki > 10000 nM T84117 CW83DK 73213196 Ki > 10000 nM T84117 C2E7QW 75201901 Ki = 9800 nM T84117 C8IDL3 75306277 Ki = 2511.89 nM T84117 C70ZVB 86221574 Ki > 10000 nM T84117 CEMZ15 118464420 Ki > 10000 nM T84117 CV2L6O 118464425 Ki > 10000 nM T84117 CFNG86 118464427 Ki > 10000 nM T84117 C7ODW3 122195524 Ki > 900 nM T84117 C4QM2E 124247485 Ki = 793 nM T84117 CTBN56 127026052 Ki = 478.63 nM T84117 CU49VE 127036186 Ki = 489.78 nM T84117 CG06BD 127036932 Ki = 354.81 nM T84117 CVW71O 127036953 Ki = 512.86 nM T84117 C50GOC 130442480 Ki = 8900 nM T84117 CM04RF 130442572 Ki = 9900 nM T84117 CY8B9L 132060743 Ki = 403 nM T84117 C7FM0U 132060763 Ki = 1242 nM T84117 CGHO19 132060770 Ki = 1666 nM T84117 CAVB41 132584404 Ki > 10000 nM T84117 CBU81N 134149168 Ki > 10000 nM T84117 C6N8GM 135367405 Ki = 890 nM T84117 C6LU0C 135367816 Ki > 10000 nM T84117 CD2TH9 135367820 Ki > 10000 nM T84117 C5AMD9 135367857 Ki = 1787 nM T84117 C8WL0I 135449090 Ki > 10000 nM T84117 C03HVY 135846955 Ki > 10000 nM T84117 CE4QG5 135846981 Ki > 10000 nM T84117 C3UB7L 135846982 Ki > 10000 nM T84117 CUKO20 136020617 Ki > 10000 nM T84117 COF0U5 136020618 Ki > 10 nM T84117 CF89JI 136030596 Ki > 10000 nM T84117 CE8GB9 136030693 Ki > 10000 nM T84117 C65VFI 136030744 Ki > 10000 nM T84117 COIX80 136054961 Ki > 10000 nM T84117 C6R4IC 136118615 Ki > 10000 nM T84117 CHWC38 136118619 Ki > 10000 nM T84117 C5UDW3 136118620 Ki > 10000 nM T84117 C8I6UN 136118621 Ki > 10000 nM T84117 CCHM67 136118657 Ki > 10000 nM T84117 C0W1TM 136118658 Ki > 10000 nM T84117 CON04G 136118728 Ki > 10000 nM T84117 COX1F8 136118729 Ki > 10000 nM T84117 C0R5PV 136118732 Ki > 10000 nM T84117 CAE39V 136188797 Ki > 10000 nM T84117 CC6OP7 136244089 Ki > 10000 nM T84117 CLAP52 136259032 Ki > 10000 nM T84117 C7KC3T 145963830 Ki = 2400 nM T84117 CHDN35 145964150 Ki > 10000 nM T84117 C1KH2E 145964159 Ki > 10000 nM T84117 C12OVL 145965034 Ki > 10000 nM T84117 C5W4LM 145965940 Ki > 10000 nM T84117 C81VUO 145967771 Ki > 10 nM T84117 CJS56K 145967795 Ki > 10000 nM T84117 CQJ5O8 145971635 Ki > 10000 nM T84117 C7BVC1 145972374 Ki = 1400 nM T84117 C79TNE 145972796 Ki > 10000 nM T84117 C6XIN0 145974114 Ki > 10000 nM T84117 CD8ZL6 145974750 Ki > 10 nM T84117 C6PH4F 145975226 Ki = 4600 nM T84117 C71CYU 145975946 Ki > 10000 nM T84117 C2TN8W 145976085 Ki > 10000 nM T84117 C6BFY7 145977338 Ki > 10000 nM T84117 C0Y6QO 145977799 Ki = 4000 nM T84117 C3BI1R 145978113 Ki > 10000 nM T84117 CQU8R0 145978665 Ki > 10000 nM T84117 C6AV9G 145978819 Ki > 10000 nM T84117 C86XQR 145988313 Ki > 10000 nM T84117 CC2G1V 146025727 Ki = 7800 nM T84117 C6P3SR 153287553 Ki > 10000 nM T84117 CV9G7Z 153287572 Ki > 10000 nM T84117 CO85KL 153287574 Ki > 10000 nM T84117 CUSA24 155519891 Ki > 10000 nM T84117 CB79ZW 155536080 Ki > 10000 nM T84117 C3N9VU 10251906 Ki > 500 nM T84117 CRKP76 136016509 Ki > 10000 nM T84117 D00CRA 1574 Ki > 10000 nM T84117 D01HRV 9847194 IC50 > 10000 nM T84117 D03DET 10287730 Ki < 10000 nM T84117 D04AZE 3277600 Ki < 100000 nM T84117 D05XGR 6918647 Ki = 1584.89 nM T84117 D07LRJ 5312149 Ki < 10000 nM T84117 D08CKM 9863250 Ki < 10000 nM T84117 D09OYA 2107 Ki > 10000 nM T84117 D09PIN 3378093 Ki > 10000 nM T84117 D09RPR 16737207 Ki > 10000 nM T84117 D09WIL 10028436 Ki < 5011.87 nM T84117 D0C5GF 6918515 Ki > 10000 nM T84117 D0CK9K 6918513 Ki = 520 nM T84117 D0F6CD 5202 Ki = 4 nM T84117 D0H7PC 6918553 Ki > 10000 nM T84117 D0H9QG 5312148 Ki < 15848.93 nM T84117 D0L5MW 181743 Ki > 10000 nM T89879 D04AIT 5280445 IC50 = 20000 nM T89879 D07EXH 359 IC50 > 200000 nM T89879 D07MGA 72281 IC50 = 8300 nM T89879 D0J9ZR 4477 IC50 = 40000 nM T89879 D0K8KX 5280343 IC50 = 8100 nM T89879 C5H9TY 14697 IC50 = 207000 nM T89879 C3I7VB 102678 IC50 = 24500 nM T89879 CL5Y4J 159516 Ki = 3100 nM T89879 CV0B7W 442027 IC50 = 49600 nM T89879 C1E2FR 442048 IC50 = 283500 nM T89879 CZ3MD8 647122 IC50 = 16100 nM T89879 C2C8QU 948801 Ki = 27500 nM T89879 CXA4P6 1265413 IC50 = 90720 nM T89879 CUD4A1 1328543 IC50 = 58350 nM T89879 C3ZP4U 2131972 Ki = 9110 nM T89879 CA1N3H 2131982 Ki = 9930 nM T89879 CKL8B2 2219105 IC50 = 29900 nM T89879 CN43XQ 2806068 IC50 = 160 nM T89879 C5J6MO 2849659 IC50 = 28800 nM T89879 CN3P7A 2911959 IC50 = 74500 nM T89879 CZDG23 2947583 IC50 = 186000 nM T89879 CBIP72 2986413 IC50 = 76700 nM T89879 CCU3P7 3635406 IC50 = 2200 nM T89879 CZF0R5 4004950 IC50 = 500 nM T89879 C3AN7C 4117477 IC50 = 1180 nM T89879 CS2WB7 4236803 IC50 = 29800 nM T89879 C0AW3N 4378077 IC50 = 13860 nM T89879 CO3Y0T 4614896 IC50 = 9910 nM T89879 CY68ZT 4788586 IC50 = 940 nM T89879 CTR4Q1 5320532 IC50 = 13300 nM T89879 CVG47I 5958938 IC50 = 10500 nM T89879 CD8ZT2 6026688 IC50 > 50000 nM T89879 C3LZX9 8027611 IC50 = 12660 nM T89879 CJ4C5K 9180583 IC50 = 10800 nM T89879 CYQ8Z4 9882716 IC50 > 50000 nM T89879 C8K2NO 10062715 IC50 = 800000 nM T89879 C49CMU 10411574 IC50 = 21700 nM T89879 C6GN2F 11642725 IC50 = 870000 nM T89879 CHYP53 12310492 IC50 = 233400 nM T89879 C65EOH 15949840 IC50 = 7500 nM T89879 C9V8EM 15956553 IC50 = 300000 nM T89879 C3WYR4 16061499 IC50 = 2000 nM T89879 CTO43V 16085283 Ki = 116000 nM T89879 CU35DQ 21582568 IC50 = 220800 nM T89879 CN45FL 23427055 IC50 = 164700 nM T89879 CK3AF8 25256829 IC50 = 5400 nM T89879 C2SZ7L 42624533 IC50 = 14000 nM T89879 CYP8V1 44404067 IC50 > 50000 nM T89879 CD20PF 44433696 IC50 = 80000 nM T89879 CI4P2V 44433697 IC50 = 10000 nM T89879 CW7B0J 44433698 IC50 = 15000 nM T89879 C8DWL3 44433699 IC50 = 200000 nM T89879 C0ZPE2 44517748 IC50 = 2700 nM T89879 C0OH2T 44584893 IC50 = 5400 nM T89879 C0NZ5E 44584944 IC50 = 7300 nM T89879 CT70DZ 44590821 IC50 = 22500 nM T89879 C0SW2K 45266425 IC50 = 2500 nM T89879 C5WBP2 45266482 IC50 = 3800 nM T89879 CA4K8F 45266488 IC50 = 6600 nM T89879 C3BHZ4 45268445 IC50 > 50000 nM T89879 CC05NI 45268452 IC50 = 15400 nM T89879 C6QD9E 45269292 IC50 > 50000 nM T89879 CY7RV4 45269761 Ki = 21000 nM T89879 CO80TH 45269762 Ki = 297000 nM T89879 CU34ZK 45269763 Ki = 584000 nM T89879 C9P3LZ 45269764 Ki = 478000 nM T89879 CXS19V 45269765 Ki = 45200 nM T89879 C3DY4T 45270971 IC50 > 50000 nM T89879 CR4WA8 45270979 IC50 = 20900 nM T89879 CM78GO 45271412 Ki = 462000 nM T89879 CC90BU 45271826 IC50 = 5200 nM T89879 C0B6KX 45271831 IC50 = 9300 nM T89879 CN85IQ 45271832 IC50 = 8100 nM T89879 C7IF2O 45272299 Ki = 363000 nM T89879 CZRV73 45272304 Ki = 34100 nM T89879 CGV14L 45272305 Ki = 112000 nM T89879 CVTL97 45272306 Ki = 2200 nM T89879 CAM89I 45273174 Ki = 135000 nM T89879 CZT67B 45273179 Ki = 614000 nM T89879 CHF4M5 45273180 Ki = 49300 nM T89879 CND1R3 45273184 Ki = 159000 nM T89879 C0V5WT 45273625 IC50 > 50000 nM T89879 C6OE7V 46784066 IC50 = 28300 nM T89879 C6LH5I 46881919 Ki = 800 nM T89879 CI2FO1 49870840 IC50 = 5500 nM T89879 CF2D0I 49870841 IC50 = 8400 nM T89879 CM52SZ 49870842 IC50 = 6800 nM T89879 C8Q2CZ 50885062 IC50 > 50000 nM T89879 CJ6KV7 52941131 IC50 = 13900 nM T89879 C8M2QD 52943127 IC50 = 24300 nM T89879 CQ84MD 52945913 IC50 = 12000 nM T89879 CJ1LG2 52945915 IC50 = 42000 nM T89879 CZ35DX 52945977 IC50 = 128900 nM T89879 CAB1Y3 52946772 IC50 = 163200 nM T89879 CO4R1B 52947200 IC50 = 18000 nM T89879 CC4X1O 52948928 IC50 = 137700 nM T89879 CMG4U7 52949213 IC50 = 10800 nM T89879 C0X5BL 58589722 IC50 = 76740 nM T89879 CY3CL6 71544384 IC50 = 610 nM T89879 CV3P2U 71544385 IC50 = 230 nM T89879 CJS60O 71571220 IC50 = 49000 nM T89879 C1AY0M 71571221 IC50 = 49000 nM T89879 CY21XB 71571222 IC50 = 4600 nM T89879 C1DX9H 71571223 IC50 = 39000 nM T89879 CKE2C3 73056463 IC50 > 100000 nM T89879 C9S8ZH 73056464 IC50 > 100000 nM T89879 CK9OI0 73056465 IC50 = 31710 nM T89879 C4D8LK 73056466 IC50 = 32080 nM T89879 CRY86G 73056467 IC50 = 34910 nM T89879 C3VS4F 73056760 IC50 = 10070 nM T89879 CYH1F4 73056761 IC50 = 51330 nM T89879 C2CRZ8 73056762 IC50 = 2250 nM T89879 CD4YR3 73056763 IC50 = 11830 nM T89879 C3P2OZ 73056764 IC50 = 67200 nM T89879 C1H8PX 73056765 IC50 = 82910 nM T89879 C8JO7B 73056766 IC50 = 13860 nM T89879 CCYE63 73057087 IC50 = 5520 nM T89879 C54JWM 73057088 IC50 = 39870 nM T89879 C8RBU6 73057089 IC50 = 1040 nM T89879 CEBH65 73057090 IC50 = 1690 nM T89879 C8M2DX 73057091 IC50 = 17820 nM T89879 CQ42AZ 73057092 IC50 = 2820 nM T89879 CPLJ64 73057388 IC50 = 4700 nM T89879 CIN5V0 76320984 IC50 = 4300 nM T89879 C05AYV 102341658 IC50 = 16400 nM T89879 C8S3CR 102341659 IC50 = 37500 nM T89879 C2G9CP 127043455 IC50 = 20200 nM T89879 CVZ4I3 127043641 IC50 = 6000 nM T89879 C7BST4 127043642 IC50 = 5800 nM T89879 CGO01F 127043643 IC50 > 50000 nM T89879 C2TU5A 127043644 IC50 = 6400 nM T89879 C0Y9IT 127043645 IC50 = 41200 nM T89879 CF3B1Z 127045220 IC50 = 11700 nM T89879 CIXJ94 127045221 IC50 = 8600 nM T89879 CQ1CT5 127045222 IC50 = 18700 nM T89879 CKRX04 127045227 IC50 = 30700 nM T89879 CDZ2E1 127045228 IC50 > 50000 nM T89879 CG3E9B 127045229 IC50 = 6700 nM T89879 CG6VR3 127045386 IC50 = 15700 nM T89879 CK9JE3 127045387 IC50 > 50000 nM T89879 CY1E4Z 127045392 IC50 > 50000 nM T89879 CK5PA4 127045393 IC50 = 44700 nM T89879 C34TWD 127045394 IC50 > 50000 nM T89879 C97MQC 127048409 IC50 = 20000 nM T89879 C41VRM 127048410 IC50 = 7500 nM T89879 CZ0B1R 127052510 IC50 = 10000 nM T89879 CRW05E 127052511 IC50 > 50000 nM T89879 CC3TX0 127052512 Ki = 72000 nM T89879 CIQ1U9 127052513 Ki = 41000 nM T89879 CI13JZ 135452883 IC50 = 10000 nM T89879 CG1KW5 135470831 IC50 = 77090 nM T89879 CH4Q6A 145964401 IC50 = 5500 nM T89879 CHU61S 145964420 IC50 = 42100 nM T89879 C6YCA8 145964710 IC50 = 28800 nM T89879 CV6F7L 145966788 IC50 = 2100 nM T89879 CBWX17 145967285 IC50 = 4300 nM T89879 COR9X3 145972736 IC50 = 3900 nM T89879 CQ0M2X 145972809 IC50 = 4100 nM T89879 CF95RZ 145972878 IC50 = 3200 nM T89879 CXI0D1 145975081 IC50 = 6300 nM T89879 CG84ZR 145975487 IC50 = 5100 nM T89879 C91FOT 145976006 IC50 = 5200 nM T89879 C3F4UH 145978039 IC50 = 8800 nM T89879 CL7FB0 2919450 IC50 = 62790 nM T89879 D00RIX 5280443 IC50 = 280800 nM T89879 D01XMM 4117383 IC50 = 4450 nM T89879 D08MZY 145937 Ki = 8200 nM T89879 D08UYP 3008868 Ki = 2400 nM T89879 D09BUG 10207 IC50 = 132000 nM T89879 D0L7AT 10480940 Ki = 19300 nM T89879 D0S0BN 130976 Ki = 10600 nM T89879 D0SY2M 5281708 IC50 = 105000 nM T89879 D0UQ6U 10569 IC50 = 189100 nM T89879 D0WA9S 10429214 IC50 = 146500 nM T88752 C43DAY 68635 IC50 = 4600 nM T88752 C5KW4H 72311 IC50 = 7000 nM T88752 CYUH56 363208 IC50 = 31000 nM T88752 CWJ43S 443767 IC50 = 34000 nM T88752 CORM47 1849091 IC50 = 21300 nM T88752 C9N5XB 2026662 IC50 = 8700 nM T88752 CD8BS4 2999946 IC50 = 46100 nM T88752 CYZ0U7 4891910 IC50 = 5300 nM T88752 CAK90T 4893331 IC50 = 27900 nM T88752 CU8LQ0 4893774 IC50 = 24200 nM T88752 CF9QP2 9076354 IC50 = 24100 nM T88752 CT8RA9 9099810 IC50 = 57200 nM T88752 CK7N4D 9880653 IC50 = 2700 nM T88752 CD57RY 24344410 IC50 = 28300 nM T88752 CN3Y9K 25138381 IC50 = 9300 nM T88752 CDU76N 25164618 IC50 = 54000 nM T88752 C4OP0C 25165019 IC50 = 58000 nM T88752 C51DAH 45272995 IC50 = 12200 nM T88752 CP57CD 45483073 IC50 = 13000 nM T88752 CURM73 51031035 IC50 = 1100 nM T88752 C0EQA8 90655048 IC50 = 95000 nM T88752 C1KBS9 135431654 IC50 = 1800 nM T88752 C9PY6U 135959764 IC50 = 37000 nM T12581 CS1QX6 125545 EC50 = 210 nM T12581 CYPF58 443266 IC50 = 430 nM T12581 CVJZ65 12068910 IC50 = 6.1 nM T12581 C7R4XW 44458634 IC50 = 44 nM T12581 D0MH9X 107758 IC50 = 2.9 nM T12581 D0W1GH 121920 IC50 = 620 nM T84133 D05MQK 110635 IC50 > 10000 nM T84133 D06BCB 443955 IC50 > 10000 nM T84133 D0C9SY 135400189 IC50 = 790 nM T84133 D0F9GE 3108 Ki = 1000 nM T84133 D0NJ3V 4680 IC50 = 21 nM T84133 D0Z7ZM 135398744 IC50 = 3100 nM T84133 D01LCC 17754438 IC50 = 2700 nM T84133 D0EY0A 42636350 IC50 = 5500 nM T84133 D0OH2W 11581936 IC50 = 0.37 nM T84133 D0T5PO 5092 IC50 > 16000 nM T84133 D0X0PP 59351313 IC50 = 0.1 nM T84133 D01ITP 71295652 IC50 = 9 nM T84133 D03GTM 118485599 IC50 > 10000 nM T84133 D05VBJ 71295299 IC50 = 1760 nM T84133 D07EUB 46200734 IC50 = 9.83 nM T84133 D09BDD 56933838 IC50 = 506 nM T84133 D0J1LK 118485649 IC50 = 1200 nM T84133 D0WS3T 72706254 IC50 = 690 nM T84133 D00YPW 135399235 IC50 = 22000 nM T84133 D01FXD 9802841 IC50 > 10000 nM T84133 C0NP3E 7195 Ki = 500000 nM T84133 C4IQ1D 11829 Ki = 590000 nM T84133 CX06SW 11830 Ki = 94000 nM T84133 CBU72A 13021 Ki = 1300000 nM T84133 C67CJL 29872 Ki = 210000 nM T84133 CBIG84 66593 Ki = 500000 nM T84133 CIN2O4 67432 Ki = 410000 nM T84133 CL51WY 76081 Ki = 16000 nM T84133 C03JPW 76143 Ki = 1200000 nM T84133 C3YI1T 217632 Ki > 1000 nM T84133 C09RTL 243166 Ki = 300000 nM T84133 CG5QY2 305345 IC50 > 1000 nM T84133 C9LH4S 371187 IC50 = 48.8 nM T84133 C1B6ZL 662965 IC50 > 50000 nM T84133 CN9WF3 700124 IC50 = 851000 nM T84133 CM1XC0 735871 IC50 < 10000 nM T84133 CA5R2Z 866356 IC50 > 10000 nM T84133 CRW0V2 1122713 IC50 = 35 nM T84133 CHPF20 1188002 IC50 = 39 nM T84133 CNZ6L4 1366773 Ki = 87 nM T84133 CR94IK 1415219 IC50 = 210 nM T84133 C8JLO0 2243267 IC50 = 3500 nM T84133 C38ELQ 2776174 Ki = 940000 nM T84133 C7MYP8 2884317 IC50 = 68 nM T84133 CCL7M3 3685273 IC50 = 1000 nM T84133 CK12OT 3814427 IC50 = 84 nM T84133 CZ71SC 4080937 IC50 > 10000 nM T84133 CF95QS 4195078 IC50 = 3000 nM T84133 CVQ8G9 4259342 IC50 = 380 nM T84133 CW7AM9 4458268 IC50 = 4500 nM T84133 C2LMB4 5151485 IC50 = 310 nM T84133 CMK39Q 10553487 IC50 > 10000 nM T84133 C4BC0Z 10680968 IC50 = 1800 nM T84133 CF4SN3 11074154 Ki = 24000 nM T84133 C45VZC 11438405 IC50 > 16000 nM T84133 CIM6H8 11504190 IC50 = 16 nM T84133 CE0XC8 11512099 IC50 = 22 nM T84133 CJH21A 11517420 IC50 = 41.5 nM T84133 CI15RY 11525659 IC50 = 7 nM T84133 CLI15E 11533673 IC50 = 120 nM T84133 C4ZYH9 11547485 IC50 = 2200 nM T84133 CI95DB 11576116 IC50 = 6 nM T84133 C53ZEH 11590899 IC50 = 3 nM T84133 C3G1BO 11604203 IC50 = 0.28 nM T84133 C5S1WA 11613446 IC50 = 3 nM T84133 CQ6Z7B 11634505 IC50 = 4 nM T84133 CS3J8Z 11635020 IC50 = 2 nM T84133 C6GY9D 11635241 IC50 = 1900 nM T84133 C40YUX 11637556 IC50 = 16300 nM T84133 CB2G3L 11641069 IC50 = 2 nM T84133 C2J7OE 11641566 IC50 = 34 nM T84133 CU2RN6 11648276 IC50 = 0.3 nM T84133 C94GTK 11655421 IC50 = 4 nM T84133 CR8CQ7 11669507 IC50 = 0.29 nM T84133 C3XYS6 11698194 IC50 = 6 nM T84133 COU75F 11710344 IC50 = 3 nM T84133 CC1S6V 11720710 IC50 = 2 nM T84133 CA26IK 11742611 IC50 > 10000 nM T84133 CL6F4C 11955614 Ki = 4 nM T84133 CUK49V 11988837 Ki = 2700 nM T84133 CFIO49 11988967 Ki = 7900 nM T84133 C2D0NG 11989101 Ki = 5400 nM T84133 C65ABT 11989102 Ki = 19000 nM T84133 CY20HE 14943631 IC50 = 890 nM T84133 CSX70H 15991588 Ki = 12 nM T84133 C08TUE 16102593 Ki = 811 nM T84133 C7GDQ8 16102594 Ki = 240 nM T84133 CHAL10 16102596 Ki = 130 nM T84133 C6Z7GM 16102598 Ki = 54 nM T84133 C4JVF5 16102599 Ki = 136 nM T84133 CMR3A7 16102600 Ki = 68 nM T84133 CX1B4L 16102601 Ki = 44 nM T84133 CC0DP8 16102602 Ki = 123 nM T84133 CLH34A 16102603 Ki = 112 nM T84133 CK06QM 16102604 Ki = 210 nM T84133 C4TH8R 16102605 Ki = 17 nM T84133 C6X1VB 16102606 Ki = 18 nM T84133 C04SBT 16102607 Ki = 19 nM T84133 C9IK5Y 16102620 Ki = 326 nM T84133 CL6Y7J 16102621 Ki = 198 nM T84133 CNAW90 16102622 Ki = 56 nM T84133 C1GD3A 16102623 Ki = 100 nM T84133 CA52VZ 16102625 Ki = 94 nM T84133 CH25WX 16102626 Ki = 67 nM T84133 C5V1LM 16102627 Ki = 128 nM T84133 CC21RZ 16102628 Ki = 18 nM T84133 C5SN6Y 16102629 Ki = 12 nM T84133 C3S2KA 16102630 Ki = 12 nM T84133 C9XNR3 16419285 IC50 = 2400 nM T84133 C1L2MA 16582132 IC50 = 2500 nM T84133 COG39H 16727125 IC50 = 1500 nM T84133 C0MA2Z 17437959 IC50 = 15 nM T84133 C6J4OB 17454842 IC50 = 110 nM T84133 CXFT59 17757146 IC50 = 823 nM T84133 C1PZ8C 18734933 IC50 > 16000 nM T84133 C25GCV 19935268 Ki = 380000 nM T84133 CGJH45 21002944 IC50 = 1800 nM T84133 C7YT4G 21259157 IC50 = 324000 nM T84133 CW96SI 23624262 IC50 = 7 nM T84133 CJ0ZF1 24180492 IC50 = 430 nM T84133 C8MU9Q 24745788 IC50 = 21.4 nM T84133 CW2US9 24746467 IC50 = 125 nM T84133 C6LV1F 24802716 IC50 = 12.4 nM T84133 C9WGI4 24802717 IC50 = 7.28 nM T84133 CC25EQ 24802718 IC50 = 15.7 nM T84133 COM21S 24802719 IC50 = 81.2 nM T84133 C08NUH 24802721 IC50 = 51.3 nM T84133 C2OB3S 24802722 IC50 = 2.84 nM T84133 C7NVY6 24802884 IC50 = 223 nM T84133 C7CAQ3 24802885 IC50 = 116 nM T84133 C01PNE 24802891 IC50 = 8.32 nM T84133 C2QV8Z 24803049 IC50 = 32.5 nM T84133 CE4SQ3 24803050 IC50 = 25.1 nM T84133 CGT60I 24803051 IC50 = 13.2 nM T84133 COTR52 24803223 IC50 = 22.9 nM T84133 C3NKC1 24803224 IC50 = 206 nM T84133 CDEK56 24803227 IC50 = 535 nM T84133 CC6XU8 24803383 IC50 = 55.4 nM T84133 C67TRL 24803384 IC50 = 381 nM T84133 CVZ1G5 24803385 IC50 = 15.3 nM T84133 CO6ZN3 24803386 IC50 = 39.2 nM T84133 C9DSN4 24803387 IC50 = 64.7 nM T84133 C2TR8E 24803388 IC50 = 53.4 nM T84133 CN7GJ6 24803389 IC50 = 617 nM T84133 CI54GC 24803543 IC50 = 132 nM T84133 CFG52I 24804535 IC50 = 24.8 nM T84133 C0GY4W 24804536 IC50 = 92.2 nM T84133 CJ1U3Z 24804537 IC50 = 63 nM T84133 C4O0IX 24804538 IC50 = 270 nM T84133 CJ40AC 24804539 IC50 = 2270 nM T84133 CKR97Z 24804540 IC50 = 731 nM T84133 C5XFP1 24804699 IC50 = 149 nM T84133 C05DQY 24804701 IC50 = 391 nM T84133 CFC7X5 24804871 IC50 = 383 nM T84133 CZ4R9U 24805030 IC50 = 962 nM T84133 C8B5LM 24805034 IC50 = 617 nM T84133 CS0I7F 24805035 IC50 = 209 nM T84133 CE6QM4 24805036 IC50 = 2390 nM T84133 C76DWZ 24805199 IC50 = 10.9 nM T84133 CXB7H2 24805200 IC50 = 36.4 nM T84133 C07XUR 24805202 IC50 = 23.3 nM T84133 C6GIQ3 24805203 IC50 = 89.6 nM T84133 C10ADY 24805204 IC50 = 284 nM T84133 C79SXK 24805205 IC50 = 33.9 nM T84133 C20VHK 24871823 IC50 = 85 nM T84133 C0E9RA 24983496 IC50 = 9.7 nM T84133 C9WX7I 25195576 IC50 = 1.5 nM T84133 CG4HU9 25195579 IC50 = 7 nM T84133 CL1S8F 25195685 IC50 = 1.1 nM T84133 C0R2EF 25195686 IC50 = 17.3 nM T84133 CL1N8C 25195687 IC50 = 16.3 nM T84133 CQ64SM 25196602 IC50 = 4.9 nM T84133 CGZP65 25196603 IC50 = 13.2 nM T84133 CD35KE 25196606 IC50 = 1.2 nM T84133 C9BQI5 25196607 IC50 = 2.6 nM T84133 C9GIO4 25196715 IC50 = 3.2 nM T84133 CV0F2B 25196716 IC50 = 5.8 nM T84133 C4J0YD 25196719 IC50 = 1.52 nM T84133 CAR7F0 25197023 IC50 = 1.3 nM T84133 C64KEG 25218869 IC50 = 400 nM T84133 C4I8XH 42623946 IC50 = 472 nM T84133 CD4NM7 42623948 IC50 = 175 nM T84133 C14KMP 42624027 IC50 = 1050 nM T84133 CEJ67W 42624216 IC50 = 246 nM T84133 CJ6UR1 42624218 IC50 = 482 nM T84133 CMI41E 42624219 IC50 = 146 nM T84133 CS7RC9 42629350 IC50 = 13.3 nM T84133 C7SGR9 42629353 IC50 = 14.4 nM T84133 C9CE2J 42629699 IC50 = 13.9 nM T84133 CP9TE3 42629700 IC50 = 14.9 nM T84133 CICF39 42629702 IC50 = 11 nM T84133 CIFO36 42629821 IC50 = 65.3 nM T84133 CMIX45 42629822 IC50 = 173 nM T84133 CM3X9S 42629827 IC50 = 7.4 nM T84133 C29JFA 42629944 IC50 = 186 nM T84133 CQN26J 42629945 IC50 = 7.4 nM T84133 CRX87A 42629953 IC50 = 11 nM T84133 C6O5FX 42630062 IC50 = 1.8 nM T84133 CR2VK6 42630063 IC50 = 24 nM T84133 C1A4UY 42630064 IC50 = 20.5 nM T84133 CWT8E7 42630065 IC50 = 14.4 nM T84133 C70YVS 42630068 IC50 = 79.5 nM T84133 CTS74L 42630069 IC50 = 22 nM T84133 C3P1XN 42630071 IC50 = 3.9 nM T84133 C2O1WH 42630072 IC50 = 11.7 nM T84133 CGU0S3 42630073 IC50 = 1.5 nM T84133 C71ZNR 42630180 IC50 = 2.8 nM T84133 C7T8DM 42630184 IC50 = 46 nM T84133 C9UZW3 42630188 IC50 = 2.9 nM T84133 CX9ZT6 42630190 IC50 = 2 nM T84133 C4RHY0 42630191 IC50 = 0.7 nM T84133 CT6RS9 42630192 IC50 = 0.55 nM T84133 CYLS05 42630193 IC50 = 0.35 nM T84133 C7J0PY 42630314 IC50 = 1.5 nM T84133 CJC7B8 42630315 IC50 = 0.85 nM T84133 CCPV45 42630316 IC50 = 63.9 nM T84133 CYZL43 42630317 IC50 = 0.5 nM T84133 CH42OZ 42630318 IC50 = 0.2 nM T84133 C7X5AH 42630437 IC50 = 0.14 nM T84133 C8L7XT 42630438 IC50 = 7.5 nM T84133 C0ZFQ8 42630439 IC50 = 102 nM T84133 C5IVS3 42630440 IC50 = 1.9 nM T84133 CKE04L 42630684 IC50 = 9.62 nM T84133 CGV5A0 42630796 IC50 = 6 nM T84133 C18ZNC 42630799 IC50 = 21.4 nM T84133 C5Q0IN 42647289 IC50 = 388 nM T84133 CNIE98 44143458 IC50 = 632 nM T84133 CW8OB3 44243146 Ki = 1 nM T84133 CE8CL6 44440359 IC50 = 140 nM T84133 CWV38B 44440363 IC50 = 45 nM T84133 C6XB2I 44440367 IC50 = 30 nM T84133 C4Q1AZ 44440369 IC50 = 35 nM T84133 CG04FU 44440370 IC50 = 35 nM T84133 COCF81 44440373 IC50 = 7 nM T84133 CR25KM 44440389 IC50 = 5 nM T84133 CMAD80 44440391 IC50 = 0.3 nM T84133 C4RTA8 44440392 IC50 = 10 nM T84133 C9G1QE 44440395 IC50 = 1 nM T84133 CT7Q2I 44440397 IC50 = 4 nM T84133 CI87NE 44440399 IC50 = 2 nM T84133 CS07MP 44440400 IC50 = 18 nM T84133 CH0KB2 44440401 IC50 = 3 nM T84133 CF80NI 44440403 IC50 = 6 nM T84133 CJQP98 44440404 IC50 = 21 nM T84133 CS6W5I 44440405 IC50 = 1900 nM T84133 CM0PA2 44440406 IC50 > 4000 nM T84133 CVR47J 44440407 IC50 = 100 nM T84133 CX0LW3 44440408 IC50 = 18 nM T84133 CVK5U4 44440409 IC50 = 120 nM T84133 CJCX12 44440410 IC50 = 160 nM T84133 C4UD9G 44440415 IC50 = 79 nM T84133 C8JDH7 44440416 IC50 = 4000 nM T84133 CA0E7D 44440418 IC50 = 1300 nM T84133 C1NZE3 44441802 IC50 = 2800 nM T84133 CM13IX 44441825 IC50 = 130 nM T84133 CSD1Q8 44441827 IC50 = 1100 nM T84133 CG49SA 44441829 IC50 = 600 nM T84133 C8FK0V 44441831 IC50 = 120 nM T84133 CTI03C 44441833 IC50 = 20 nM T84133 CZYW49 44441837 IC50 = 760 nM T84133 CQ0N7Y 44441840 IC50 = 1700 nM T84133 C98UBL 44452447 Ki = 185 nM T84133 CPOZ04 44452603 Ki = 171 nM T84133 CK9NU0 44537944 IC50 = 7.2 nM T84133 CUO2D3 44539913 IC50 < 50 nM T84133 CCVO04 44546588 IC50 < 50 nM T84133 CS2A4J 44547515 IC50 = 0.32 nM T84133 CY41QP 44547965 IC50 = 0.32 nM T84133 C7GNE3 44548113 IC50 = 67 nM T84133 CGP02T 44555440 IC50 < 50 nM T84133 CDQP73 44608934 IC50 = 7.2 nM T84133 CM83YD 46174637 IC50 = 0.0033 nM T84133 CI68SV 46178283 IC50 = 0.44 nM T84133 C6LZJ3 46185994 IC50 < 50 nM T84133 CC0OM2 46185995 IC50 < 50 nM T84133 C0D2MN 46186792 IC50 = 13.1 nM T84133 CR1K5E 46198523 IC50 = 9.6 nM T84133 C58BSW 46198541 IC50 = 2430 nM T84133 C1BIJ2 46198546 IC50 = 388 nM T84133 CC42ER 46198694 IC50 = 45.5 nM T84133 C0WRO9 46198713 IC50 = 45.9 nM T84133 CON1M4 46199019 IC50 = 91.3 nM T84133 C5AND7 46199167 IC50 = 114 nM T84133 CKX1A6 46199301 IC50 = 23.7 nM T84133 CZU0H7 46199329 IC50 = 51.5 nM T84133 CD9LN1 46199458 IC50 = 77.2 nM T84133 CXG34R 46199487 IC50 = 47.6 nM T84133 CAL85J 46199794 IC50 = 12.4 nM T84133 CZF5C0 46199795 IC50 = 42.4 nM T84133 CI9EA4 46199799 IC50 = 10.1 nM T84133 C26RJV 46200090 IC50 = 3.3 nM T84133 C5WND9 46200233 IC50 = 1.48 nM T84133 CKIC45 46200238 IC50 = 4.16 nM T84133 CS46AE 46200399 IC50 = 2.06 nM T84133 C1S3BK 46200706 IC50 = 1.53 nM T84133 C4P5QJ 46200709 IC50 = 2.41 nM T84133 CV8Y6W 46200711 IC50 = 3.99 nM T84133 CK1N4X 46200728 IC50 = 15 nM T84133 CH9FU8 46200877 IC50 = 8.33 nM T84133 CEZ3V4 46200878 IC50 = 9.43 nM T84133 C10HQS 46207696 IC50 < 25 nM T84133 C5N9FO 46207938 IC50 = 4.5 nM T84133 CF8UT3 46207939 IC50 = 24.4 nM T84133 CNHS37 46208071 IC50 = 2.8 nM T84133 COGX29 46208072 IC50 = 4.1 nM T84133 CRBA01 46208073 IC50 = 7.2 nM T84133 CJKH84 46208209 IC50 = 20.6 nM T84133 CIJ62X 46208210 IC50 = 5.1 nM T84133 CRXN04 46208214 IC50 = 5.1 nM T84133 C6IRP8 46208470 IC50 = 1.7 nM T84133 CF6Z5P 46208937 IC50 = 168 nM T84133 CAO2U6 46208939 IC50 = 1.1 nM T84133 C8DY5G 46209045 IC50 = 4.3 nM T84133 C36XLQ 46209046 IC50 = 4.2 nM T84133 C2Q4YT 46209162 IC50 = 138 nM T84133 CJOE41 46209386 IC50 = 0.199 nM T84133 C3P4SJ 46209520 IC50 = 1 nM T84133 C7ZY8O 46219578 IC50 = 14 nM T84133 C4UL5T 46238926 IC50 < 100 nM T84133 CU73QW 46238927 Ki = 130 nM T84133 CB9S1L 46239023 Ki = 3 nM T84133 C0V6EL 46239024 Ki = 280 nM T84133 C1HNK7 46239025 IC50 < 100 nM T84133 CYQ09Z 46239122 Ki = 5 nM T84133 CH8B1X 46239123 Ki = 15 nM T84133 C8WI1G 46239124 Ki = 29 nM T84133 CLG7K1 46239125 Ki = 14 nM T84133 CAE91W 46239126 Ki = 409 nM T84133 CV5DO7 46239228 Ki = 52 nM T84133 CED8X2 46239234 Ki = 3.3 nM T84133 CZQ5T9 46239329 Ki = 1 nM T84133 C7N8FR 46239331 Ki = 202 nM T84133 CIEM75 46239333 Ki = 871 nM T84133 CI7EX8 46239423 Ki = 32 nM T84133 C5IMB2 46239424 Ki = 3 nM T84133 CKR9P7 46239425 Ki = 3 nM T84133 CJB81K 46239426 Ki = 49 nM T84133 CEP91S 46239427 Ki = 24 nM T84133 CZV29L 46239429 Ki = 57 nM T84133 CZ5G3P 46239530 Ki = 30 nM T84133 C7SLP0 46239531 Ki = 0.6 nM T84133 CNI1U7 46239532 Ki = 37 nM T84133 CS64WE 46239728 Ki = 104 nM T84133 C95RNE 46239731 IC50 < 100 nM T84133 CAK37R 46239835 Ki = 70 nM T84133 CGBT01 46239836 Ki = 3.6 nM T84133 C08FHG 46239839 Ki = 41 nM T84133 CI1F5C 46239840 Ki = 11 nM T84133 C7P3HS 46239939 Ki = 23 nM T84133 C0X8CQ 46239940 Ki = 363 nM T84133 C0GJN1 46239943 Ki = 15 nM T84133 C26XVS 46240044 Ki = 12 nM T84133 C15QIP 46240135 Ki = 196 nM T84133 C8XFU6 46240137 Ki = 55 nM T84133 CO17GN 46683800 IC50 = 1300 nM T84133 CWB30P 46831671 IC50 = 81.5 nM T84133 C5C0KQ 46831672 IC50 = 486 nM T84133 C8TJ7K 46831673 IC50 = 1195 nM T84133 CY91XU 46831931 IC50 = 1.43 nM T84133 CKE4T9 46831932 IC50 = 7.33 nM T84133 C7TL2F 46831933 IC50 = 45.8 nM T84133 C8BWX3 46831934 IC50 = 285 nM T84133 C8RAC0 46831935 IC50 = 326 nM T84133 CE4JU7 46842025 IC50 > 10000 nM T84133 CR8JC2 46842169 IC50 > 10000 nM T84133 C6WM0L 46848741 IC50 = 0.79 nM T84133 CE6FK9 46848917 IC50 = 0.94 nM T84133 CJ4R0P 46849078 IC50 < 10 nM T84133 C9VW5F 46872031 IC50 = 27 nM T84133 C7QXI6 46873747 IC50 = 9 nM T84133 C3P2IN 46933992 IC50 >= 43000 nM T84133 COKU43 46937608 IC50 < 10 nM T84133 C3DH7C 49821302 IC50 = 5.7 nM T84133 C9Q6KE 49821304 IC50 = 3.5 nM T84133 CE8Y6Q 49821305 IC50 = 5.5 nM T84133 C94YDM 49821342 Ki = 6.1 nM T84133 C3WO9Y 49821343 Ki = 0.1 nM T84133 CAWZ34 49821394 IC50 = 0.05 nM T84133 C3TVS5 49821396 IC50 = 0.06 nM T84133 CHA5Z0 49821469 IC50 = 0.7 nM T84133 CL1BK9 49821500 Ki = 2 nM T84133 CD3C4H 49821501 Ki = 20 nM T84133 CE7GI8 49821502 Ki = 219 nM T84133 CHE15O 49821503 Ki = 0.072 nM T84133 C1ZGA8 49821582 Ki = 0.37 nM T84133 C1AYP0 49821627 IC50 = 0.09 nM T84133 C85AXR 49821714 IC50 = 0.8 nM T84133 CE41RK 49821911 Ki = 0.9 nM T84133 C5KU8W 49821931 Ki = 0.15 nM T84133 CEH5A1 49821987 Ki = 0.63 nM T84133 CF49WN 49821989 Ki = 0.92 nM T84133 C15XPB 49821991 Ki = 1 nM T84133 C29WPI 49822075 Ki = 135 nM T84133 C09BVO 49822155 Ki = 14 nM T84133 C0B8JE 49843464 IC50 < 10 nM T84133 C7Z0UN 50901948 Ki = 186 nM T84133 C3TR2P 50901952 Ki = 508 nM T84133 CMN05G 50901953 Ki = 31 nM T84133 CO4XK6 50901954 Ki = 861 nM T84133 C7V0OZ 50902028 Ki = 199 nM T84133 C9GT3X 50902029 Ki = 121 nM T84133 CZS03D 50902030 Ki = 29 nM T84133 C5I0LT 50902031 Ki = 101 nM T84133 CXT78Y 50902034 Ki = 40 nM T84133 C18FIN 50902113 Ki = 212 nM T84133 CPL5E6 50902114 Ki = 30 nM T84133 C6P8UV 50902116 Ki = 114 nM T84133 CK62ML 50902118 Ki = 628 nM T84133 CAD40F 50902119 Ki = 33 nM T84133 CD98UC 50902202 Ki = 32 nM T84133 CXB85R 50902203 Ki = 6.4 nM T84133 C9QLF2 50902206 Ki = 8 nM T84133 CH2Z1E 50902289 Ki = 20 nM T84133 C4HJL2 50902291 Ki = 25 nM T84133 C7EQ9Y 50902548 Ki = 10 nM T84133 C6A1IU 50902549 Ki = 8.7 nM T84133 CVM28N 50902550 Ki = 1.5 nM T84133 CN1P7Q 50902632 Ki = 4.3 nM T84133 C17RSC 50902804 IC50 < 10 nM T84133 C3Y2AV 50903255 Ki = 35 nM T84133 CDXL06 50942847 Ki = 15 nM T84133 CUI54F 50944015 Ki = 47.9 nM T84133 C6R4YN 50993785 IC50 = 12 nM T84133 C0M6XL 50993786 IC50 = 16 nM T84133 CSG76C 50993859 IC50 = 50 nM T84133 C6PQ3C 51000508 IC50 < 0.1 nM T84133 C2CK4X 51033482 IC50 = 0.2 nM T84133 CSNM30 51034710 IC50 = 0.1 nM T84133 C5Z3KH 51034712 IC50 = 0.1 nM T84133 C58OLQ 51304060 IC50 = 1300 nM T84133 C0IQM5 53232478 Ki = 17 nM T84133 CV35MO 53236526 IC50 = 1 nM T84133 CVRM83 53250985 IC50 = 6.7 nM T84133 CM48WF 53317312 IC50 = 76 nM T84133 CYBI97 53317313 IC50 = 50 nM T84133 C4YEK3 53317314 IC50 = 31 nM T84133 CJDV81 53318548 IC50 = 110 nM T84133 CLOI58 53319920 IC50 = 78 nM T84133 C3TI4S 53321175 IC50 = 83 nM T84133 CV3OG4 53322495 IC50 = 0.18 nM T84133 CBHF42 53323878 IC50 = 100 nM T84133 C40SMX 53323879 IC50 = 160 nM T84133 C9IVN4 53323880 IC50 = 16 nM T84133 C5JN2O 53323881 IC50 = 430 nM T84133 C5SY0C 53325113 IC50 = 130 nM T84133 C5XSA2 53325521 IC50 = 37 nM T84133 C8GH0Z 53326417 IC50 = 48 nM T84133 CZU82C 53326418 IC50 = 73 nM T84133 CZ48TX 53326461 IC50 = 52 nM T84133 CSD57U 53329353 IC50 < 1 nM T84133 COX9K5 53330053 IC50 = 2 nM T84133 CND92B 53363484 IC50 < 1000 nM T84133 CQL2P8 53378114 IC50 < 1000 nM T84133 CV3K8C 53467809 IC50 = 35 nM T84133 C7ZT0S 53468024 IC50 = 6 nM T84133 CX9Z8Q 53492734 IC50 < 100 nM T84133 CXCN02 54575101 IC50 < 100 nM T84133 CD5BR2 54575103 IC50 < 100 nM T84133 CX42VW 54575159 IC50 < 100 nM T84133 C94QRU 54576233 IC50 = 39 nM T84133 CHLA42 54576311 IC50 = 49 nM T84133 C6DEG8 54576313 IC50 = 58.5 nM T84133 CJF0K2 54576315 IC50 = 55 nM T84133 CNW81G 54576317 IC50 = 55 nM T84133 CA4I3X 54576449 IC50 = 15 nM T84133 C9WEO5 54576525 IC50 = 28 nM T84133 C3Y4WG 54576665 IC50 = 17 nM T84133 C4XM9U 54580514 IC50 = 14 nM T84133 CMG4F7 54580515 IC50 = 65 nM T84133 CE12AP 54581526 IC50 = 55 nM T84133 C19DVI 54581527 IC50 = 150 nM T84133 C9T4HK 54581943 IC50 = 1300 nM T84133 CAG1V9 54581955 IC50 = 1100 nM T84133 CV49PU 54582523 IC50 = 250 nM T84133 C2P3JM 54582524 IC50 > 10000 nM T84133 CMJ01N 54582525 IC50 = 120 nM T84133 C2RXU9 54582878 IC50 = 460 nM T84133 C59NEO 54582879 IC50 = 1000 nM T84133 CAL7N2 54582880 IC50 = 1900 nM T84133 C8ZDG9 54583877 IC50 = 320 nM T84133 CRY06I 54584473 IC50 = 130 nM T84133 C61CGS 54584474 IC50 = 790 nM T84133 CKBN97 54584475 IC50 = 190 nM T84133 CPG8Y9 54584829 IC50 > 10000 nM T84133 CL8N6Q 54585783 IC50 > 10000 nM T84133 C8XMH0 54585784 IC50 = 1600 nM T84133 C7GSO3 54585785 IC50 = 460 nM T84133 CRH83J 54585786 IC50 = 170 nM T84133 C8MGS6 54585797 IC50 = 2300 nM T84133 C8AI1O 54586387 IC50 = 8900 nM T84133 CCPD21 54586388 IC50 = 990 nM T84133 CKEP52 54586389 IC50 = 160 nM T84133 C7Z1YC 54586766 IC50 = 1500 nM T84133 CI4CO0 54587803 IC50 = 450 nM T84133 CFX89L 54587804 IC50 = 35 nM T84133 C0M5CY 54595731 Ki = 8700 nM T84133 CGF65A 54670110 IC50 = 29 nM T84133 CN4XU7 54670394 IC50 = 4100 nM T84133 C90ZLC 54670399 IC50 = 6.8 nM T84133 CAEJ46 54670484 IC50 = 7800 nM T84133 CSVE57 54670488 IC50 = 11000 nM T84133 C2JF8C 54670489 IC50 = 5700 nM T84133 C6AF1J 54671050 IC50 = 166000 nM T84133 CMT5R1 54671051 IC50 = 45000 nM T84133 C0UA1I 54674275 IC50 = 21.9 nM T84133 C5CZF9 54755130 IC50 < 500 nM T84133 CI91NY 54759276 IC50 = 140 nM T84133 C0K7YN 54760757 IC50 = 13.7 nM T84133 CJLD10 54769120 IC50 = 112 nM T84133 CKP39D 54769350 IC50 = 198 nM T84133 CWQ7S3 54769351 IC50 = 244 nM T84133 CR62YP 54769352 IC50 = 237 nM T84133 CVL03F 54769353 IC50 = 500 nM T84133 C97ACM 54769354 IC50 = 872 nM T84133 CX8P1B 54769355 IC50 = 248 nM T84133 C79BUR 54769575 IC50 = 303 nM T84133 CRA91G 54769784 IC50 = 469 nM T84133 CM96AK 54769785 IC50 = 246 nM T84133 CDRM84 56587975 IC50 = 12 nM T84133 CXI6G8 56596127 IC50 = 16 nM T84133 C1AC8K 56596128 IC50 = 93 nM T84133 CJ06ML 56596176 IC50 = 130 nM T84133 CI48VY 56596177 IC50 = 240 nM T84133 CJI54S 56596178 IC50 = 400 nM T84133 C7LF6A 56596179 IC50 = 170 nM T84133 C9NH1J 56596227 IC50 = 110 nM T84133 C7LPG5 56596228 IC50 = 31 nM T84133 CQY73S 56596229 IC50 = 61 nM T84133 C7G4FQ 56596230 IC50 = 250 nM T84133 C8FVQ1 56596231 IC50 = 12 nM T84133 COHX27 56648495 IC50 = 1.9 nM T84133 C4TGL7 56648496 IC50 = 4.3 nM T84133 C43WOF 56648497 IC50 = 60 nM T84133 CM3OI5 56648498 IC50 = 44 nM T84133 CM09EW 56648583 IC50 = 102 nM T84133 CIT68E 56648584 IC50 = 87 nM T84133 C9U0JW 56648585 IC50 = 114 nM T84133 C8O9PD 56648586 IC50 = 197 nM T84133 C52KXF 56648587 IC50 = 7.3 nM T84133 C9NC5E 56648588 IC50 = 18.2 nM T84133 CSZ6J1 56648589 IC50 = 14.2 nM T84133 CH6C3L 56648679 IC50 = 6.1 nM T84133 CCY79V 56648680 IC50 = 3.7 nM T84133 CL6Q1H 56648681 IC50 = 4.2 nM T84133 C4PH0I 56648682 IC50 = 73.4 nM T84133 CR0C8I 56648683 IC50 = 7.9 nM T84133 C15YZK 56648684 IC50 = 5.2 nM T84133 C9Z8TP 56648763 IC50 = 3.6 nM T84133 CNTL59 56648764 IC50 = 113 nM T84133 CT7QP0 56648765 IC50 = 158 nM T84133 CF95SJ 56648766 IC50 = 49.2 nM T84133 C0HX6Z 56648767 IC50 = 28.9 nM T84133 C85VDI 56648768 IC50 = 24.2 nM T84133 C0Y1RV 56648769 IC50 = 46 nM T84133 CNE96P 56648857 IC50 = 8.3 nM T84133 CU95MC 56648858 IC50 = 35.7 nM T84133 CX86AQ 56648859 IC50 = 7.4 nM T84133 CLV5E3 56648860 IC50 = 6.8 nM T84133 C6QG0A 56648861 IC50 = 11.4 nM T84133 CL8QN3 56648862 IC50 = 1.7 nM T84133 C16DEO 56648951 IC50 = 0.1 nM T84133 CG9DR0 56651641 IC50 = 0.08 nM T84133 CCM2A1 56654130 IC50 = 0.81 nM T84133 CPC3T4 56654131 IC50 = 0.76 nM T84133 CY04IO 56658425 IC50 = 200 nM T84133 CQZ4U7 56675681 IC50 = 262 nM T84133 CNX6T3 56834947 Ki = 14 nM T84133 C0YD3P 56928304 IC50 > 5000 nM T84133 C8RO6A 56929788 IC50 > 1000 nM T84133 CB5TR6 56949351 Ki = 0.01 nM T84133 CHL1C5 56949449 Ki = 0.02 nM T84133 C71JRF 56949451 Ki = 0.0082 nM T84133 CEU98Q 56949473 Ki = 9 nM T84133 CG0A3Z 56949475 Ki = 2 nM T84133 C9D8GO 56949508 Ki = 0.04 nM T84133 CP6AS2 56952795 Ki = 9.2 nM T84133 CZK51H 57328384 IC50 = 1 nM T84133 C0ZF1L 57328385 IC50 = 1 nM T84133 C8C1EW 57334262 Ki = 3 nM T84133 CLI7H6 57390414 Ki = 585 nM T84133 C9F7UR 57390415 Ki = 0.6 nM T84133 CWD1J3 57390416 Ki = 3.1 nM T84133 CZ2V5R 57390439 IC50 = 92.8 nM T84133 CJ0TI1 57390440 IC50 = 16.4 nM T84133 C94ZPA 57391164 Ki = 50 nM T84133 CD07RK 57391165 Ki = 2 nM T84133 CC76GU 57391166 Ki = 39 nM T84133 C4G1ZM 57391317 IC50 = 65 nM T84133 CC9N2A 57391318 IC50 = 22 nM T84133 C7T6XA 57391319 IC50 = 8 nM T84133 C9B5VW 57391320 IC50 = 67 nM T84133 C4QFY6 57392208 Ki = 550 nM T84133 C3TY1C 57392228 IC50 = 5.8 nM T84133 C31CEX 57392229 IC50 = 7.5 nM T84133 CZ09KG 57392230 IC50 = 13 nM T84133 C9TE7C 57392231 IC50 = 1.9 nM T84133 CR0GQ3 57392232 IC50 = 4 nM T84133 C4EGB7 57392860 IC50 = 12.9 nM T84133 C9JYK4 57392932 Ki = 12 nM T84133 CG2V1L 57392939 Ki = 26 nM T84133 CP0U1L 57392947 Ki = 153 nM T84133 CG3DF1 57392948 Ki = 8 nM T84133 CZ7X3C 57392949 Ki = 19 nM T84133 C7D3LX 57392950 Ki = 1200 nM T84133 C03TGV 57393096 IC50 = 561 nM T84133 C7GNB1 57393097 IC50 = 315 nM T84133 CZFH10 57393098 IC50 = 13 nM T84133 C6Q2PY 57393099 IC50 = 2 nM T84133 C2Z0ND 57393100 IC50 = 1770 nM T84133 CN0M9Y 57393928 IC50 = 6.2 nM T84133 CF1S9B 57393964 Ki = 0.5 nM T84133 C3R8KN 57393977 IC50 = 12.2 nM T84133 CW61NE 57394681 Ki = 171 nM T84133 CE36TV 57394695 Ki = 1 nM T84133 CMGZ76 57394696 Ki = 41 nM T84133 C9BMF8 57394826 IC50 = 21 nM T84133 C4NZS8 57395703 Ki = 419 nM T84133 CGZB82 57395734 IC50 = 124 nM T84133 C4WIC9 57395735 IC50 = 36.9 nM T84133 CF8UW0 57395736 IC50 = 10.9 nM T84133 CYV61E 57395737 IC50 = 18.6 nM T84133 CJ1UO3 57395738 IC50 = 2.6 nM T84133 C1MB4C 57395739 IC50 = 1.6 nM T84133 CE75UA 57396432 Ki = 2 nM T84133 C9K7YS 57396433 Ki = 4 nM T84133 CWE8N9 57396434 Ki = 21 nM T84133 CS0XU5 57396444 Ki = 353 nM T84133 C9L0ID 57396451 Ki = 9 nM T84133 C7VA8P 57396452 Ki = 229 nM T84133 C62JOU 57396592 IC50 = 746 nM T84133 CI25UB 57396593 IC50 = 27 nM T84133 CB71KN 57396814 Ki = 21 nM T84133 CTJN91 57397492 Ki = 35 nM T84133 CPI4V0 57397493 Ki = 27 nM T84133 C0TPH2 57397516 IC50 = 320 nM T84133 C5TJQ7 57397517 IC50 = 7.6 nM T84133 C5LNO0 57397518 IC50 = 40.6 nM T84133 CDWI58 57398224 Ki = 0.4 nM T84133 CG8B2K 57398367 IC50 = 144 nM T84133 C58IAE 57398368 IC50 = 97 nM T84133 CWQI09 57398380 IC50 = 608 nM T84133 CDSH51 57398573 Ki = 0.6 nM T84133 C7WH5G 57398574 Ki = 2 nM T84133 C8H2CI 57399125 IC50 = 3 nM T84133 CK85OQ 57399182 Ki = 6 nM T84133 CJT6U2 57399198 IC50 = 590 nM T84133 CU9XL6 57399199 IC50 = 4.4 nM T84133 C0LVB6 57399872 Ki = 83 nM T84133 C1U7LP 57399873 Ki = 1 nM T84133 CYC7S5 57399874 Ki = 0.2 nM T84133 CR9L0Z 57400027 IC50 = 9 nM T84133 CZAG81 57400035 IC50 = 13 nM T84133 C2GO5M 57400235 Ki = 54 nM T84133 CSE92V 57400886 IC50 = 1.8 nM T84133 CSQ5K8 57400960 IC50 = 10.1 nM T84133 CF7X2D 57400961 IC50 = 3 nM T84133 C7PY8W 57400962 IC50 = 2.4 nM T84133 CI0PX2 57401662 Ki = 804 nM T84133 C4PBS1 57401836 IC50 = 108 nM T84133 C3MB2N 57401837 IC50 = 31 nM T84133 CMS98N 57402038 Ki = 0.07 nM T84133 COMK36 57402700 Ki = 9.6 nM T84133 C09BLM 57402720 IC50 = 181 nM T84133 C6DI8T 57402721 IC50 = 24.4 nM T84133 CU14SI 57402722 IC50 = 9.7 nM T84133 C6B3IK 57403377 Ki = 0.3 nM T84133 CW54GL 57403378 Ki = 11 nM T84133 CI9A1D 57403379 Ki = 1 nM T84133 CPA3D1 57403394 Ki = 2 nM T84133 CQVZ29 57403395 Ki = 46 nM T84133 CU7OS0 57403396 Ki = 60 nM T84133 C14ASM 57403543 IC50 = 3 nM T84133 CR43CG 57403544 IC50 = 456 nM T84133 CJZ62H 57403545 IC50 = 52 nM T84133 C4EWA9 57403779 Ki = 0.06 nM T84133 C1H5LA 57403780 Ki = 10 nM T84133 C8HW7P 57523648 IC50 = 5.7 nM T84133 CZM4V5 58072466 IC50 < 10 nM T84133 CU8K2W 58074722 IC50 < 10 nM T84133 CRCT63 58368041 IC50 < 1 nM T84133 CSH3D7 58432081 IC50 < 1000 nM T84133 CFY5X9 58432151 IC50 < 1000 nM T84133 C7VFY2 58446918 IC50 = 1.9 nM T84133 C8I4YF 58547692 IC50 = 11000 nM T84133 C1ARH3 58547740 IC50 = 12000 nM T84133 CY7T1P 58547742 IC50 = 13000 nM T84133 CX1RJ5 58547786 IC50 = 29000 nM T84133 C7N2CL 58547789 IC50 = 147000 nM T84133 CV40CE 58547801 IC50 = 32000 nM T84133 C4XMB6 58547809 IC50 = 4700 nM T84133 CEB3G9 58547814 IC50 = 2.6 nM T84133 CYDO80 58547818 IC50 = 350000 nM T84133 CSAK24 58547819 IC50 = 46000 nM T84133 C08QVG 58547833 IC50 = 2.4 nM T84133 CP9N4A 58547845 IC50 = 54000 nM T84133 CFVG67 58547863 IC50 = 6500 nM T84133 CKR02G 58547875 IC50 = 43000 nM T84133 COD7Z3 58547879 IC50 = 38000 nM T84133 C2S8LJ 58547883 IC50 = 343000 nM T84133 C26PHF 58547902 IC50 = 41000 nM T84133 C02IVH 58547942 IC50 = 10300 nM T84133 C1GR4Z 58547944 IC50 = 64000 nM T84133 C57KYU 58547951 IC50 = 30000 nM T84133 CW82DY 58547956 IC50 = 36000 nM T84133 CYG43X 58548001 IC50 = 107000 nM T84133 C35JZX 58548005 IC50 = 45000 nM T84133 CUM63O 58548012 IC50 = 30000 nM T84133 CS80ZD 58548016 IC50 = 32000 nM T84133 CM8SN3 58548022 IC50 = 125000 nM T84133 CY5R2D 58548040 IC50 = 103000 nM T84133 CU85ZP 58548075 IC50 = 18000 nM T84133 CYZA38 58548077 IC50 = 6.8 nM T84133 C62WUD 58548080 IC50 = 39000 nM T84133 CCXW43 58548107 IC50 = 8500 nM T84133 CCHM36 58548113 IC50 = 38000 nM T84133 C91KHW 58548143 IC50 = 98000 nM T84133 C2IDR8 58548163 IC50 = 12 nM T84133 C4O5QX 58548370 IC50 = 31.5 nM T84133 C1GD9K 58578146 Ki < 1000 nM T84133 C2D4WV 58578164 Ki < 1000 nM T84133 CX7ZO2 58578167 Ki < 1000 nM T84133 CWX3N7 59320301 IC50 = 432 nM T84133 C7PB1U 59321218 IC50 = 53.1 nM T84133 CS32XI 59321284 IC50 = 1.48 nM T84133 C23WQA 59321310 IC50 = 7 nM T84133 CX45HS 59321315 IC50 = 0.7 nM T84133 CZ6C9L 59321318 IC50 = 5.11 nM T84133 C1OHZ0 59321339 IC50 = 1.85 nM T84133 C31ZBU 59326858 IC50 = 0.1 nM T84133 CHP92T 59326873 IC50 = 0.21 nM T84133 C16BHM 59326903 IC50 = 0.05 nM T84133 C6LF8T 59327006 IC50 = 0.1 nM T84133 CFL10E 59327126 IC50 = 45 nM T84133 C80VMG 59327176 IC50 = 0.96 nM T84133 C0EP5I 59341847 IC50 > 10000 nM T84133 CHQ28A 59341978 IC50 > 10000 nM T84133 CWF0O7 59351198 IC50 = 0.8 nM T84133 CJ0YB8 59351288 IC50 = 2.4 nM T84133 CZI6T1 59351366 IC50 = 7.4 nM T84133 CCA1H6 59351376 IC50 = 19.3 nM T84133 CX46SN 59351424 IC50 = 12.5 nM T84133 CEJX65 59370073 IC50 = 6 nM T84133 C64YEX 59373996 IC50 = 36.6 nM T84133 C2JW6Y 59436207 IC50 < 10 nM T84133 CMQH82 59453408 IC50 = 7 nM T84133 C0AFM6 60150358 IC50 = 0.28 nM T84133 CE0Q1S 60152740 IC50 > 1000 nM T84133 CJK53Q 60152741 IC50 = 45 nM T84133 CI3GJ1 66678348 Ki = 8.4 nM T84133 C6C8RD 66802145 IC50 = 4010 nM T84133 CU1SJ4 67075100 IC50 < 50 nM T84133 CC7B0L 67124352 IC50 = 13 nM T84133 C0SU4O 67257897 IC50 = 4.6 nM T84133 CF4A3M 67259323 IC50 = 0.27 nM T84133 CREP31 68014633 IC50 = 0.11 nM T84133 C9K8HT 68014634 IC50 = 0.13 nM T84133 CB04EH 68014656 IC50 = 0.22 nM T84133 CI68ER 68014850 IC50 = 170 nM T84133 CY8J3O 68181896 IC50 = 3900 nM T84133 C4ZEH9 68578314 IC50 = 1.82 nM T84133 CTJ46X 68594477 IC50 = 13.1 nM T84133 CV4X6K 68595169 IC50 = 64.5 nM T84133 C8E0XY 68596001 IC50 = 1.65 nM T84133 CJ80VI 68596013 IC50 = 13.1 nM T84133 CL2H4T 68596452 IC50 = 6.53 nM T84133 C93IHS 68596628 IC50 = 25.4 nM T84133 CDZ01B 68596639 IC50 = 3.55 nM T84133 C1CD9S 68596902 IC50 = 0.85 nM T84133 C7PCW0 68597211 IC50 = 9.11 nM T84133 CGJB21 68597401 IC50 = 11.7 nM T84133 CHK4S0 68597804 IC50 = 7.84 nM T84133 C10TGO 68598825 IC50 = 7.2 nM T84133 C8OD2Z 68853786 IC50 = 5.52 nM T84133 C3THF9 69568791 IC50 = 1.7 nM T84133 CFS2Z3 69569103 IC50 = 438 nM T84133 C15RXG 70169344 IC50 < 100 nM T84133 CBL8K3 70643905 Ki < 1000 nM T84133 CFPY14 70648748 IC50 < 500 nM T84133 COI2P3 70679302 IC50 = 0.097 nM T84133 CU9GQ0 70681149 Ki = 26 nM T84133 CIB7J9 70681150 Ki = 264 nM T84133 CNLD61 70681151 Ki = 183 nM T84133 CI9G8L 70683261 Ki = 3.8 nM T84133 COB1T8 70683262 Ki = 240 nM T84133 CAB45C 70684642 IC50 = 0.8 nM T84133 C6BN5J 70685361 Ki = 40 nM T84133 CM3OP8 70686796 IC50 = 5.13 nM T84133 CHBT91 70686797 IC50 = 3.35 nM T84133 CF6O3T 70687501 Ki = 6.6 nM T84133 CX6J1I 70695878 Ki = 12 nM T84133 CIBQ16 70810145 IC50 < 10 nM T84133 CC43LF 71074083 IC50 = 0.062 nM T84133 C4P0XT 71092344 IC50 = 810 nM T84133 C6DAG4 71092519 IC50 = 4030 nM T84133 CLU1S6 71151948 IC50 = 33 nM T84133 C7WD8I 71151969 IC50 = 0.1 nM T84133 C34XNL 71151981 IC50 = 20 nM T84133 C82AUP 71152059 IC50 = 20 nM T84133 C5VUO9 71152240 IC50 = 41 nM T84133 CY3RW6 71152297 IC50 = 29 nM T84133 C1M0EN 71153110 IC50 = 33 nM T84133 CZ4B9M 71153166 IC50 = 0.16 nM T84133 CG9C3J 71153201 IC50 = 29 nM T84133 C74BDZ 71153260 IC50 = 20 nM T84133 CYC05R 71153264 IC50 = 0.16 nM T84133 CCY3I0 71153278 IC50 = 41 nM T84133 CH51WI 71153284 IC50 = 33 nM T84133 C40HNF 71153309 IC50 = 29 nM T84133 C9GR3L 71153436 IC50 = 33 nM T84133 CZN5H8 71450204 IC50 = 0.34 nM T84133 CDJQ59 71450205 Ki < 1000 nM T84133 C8FEU2 71450432 Ki = 63 nM T84133 C4K1BM 71450433 Ki = 0.6 nM T84133 C8SXU3 71450486 Ki = 868 nM T84133 C2WZ8K 71450487 Ki = 156 nM T84133 CKAJ45 71450488 Ki = 864 nM T84133 CR5NQ6 71450591 IC50 = 0.941 nM T84133 CGD56M 71450592 IC50 = 6210 nM T84133 C06PTK 71452031 IC50 = 5.3 nM T84133 C06EHV 71452032 Ki = 2.19 nM T84133 CD50FS 71452033 IC50 = 3.3 nM T84133 CY6FZ1 71452252 Ki = 247 nM T84133 C1EFD6 71452326 Ki = 117 nM T84133 C9ADT4 71452327 Ki = 94 nM T84133 CZ1YN2 71452430 IC50 = 0.056 nM T84133 CI1M8Q 71452431 IC50 = 2.82 nM T84133 C6C2JD 71453832 IC50 = 0.89 nM T84133 CL6AT2 71454111 Ki = 186 nM T84133 CM6I9V 71454112 Ki = 500 nM T84133 C98ZEN 71454113 Ki = 4340 nM T84133 CX5D2O 71454197 IC50 = 422 nM T84133 C3EW1B 71455564 Ki < 1000 nM T84133 CR7Z6K 71455565 Ki < 1000 nM T84133 C5SH1U 71455566 IC50 = 0.61 nM T84133 CE3T7F 71455795 Ki = 1 nM T84133 C1JK6L 71455843 Ki = 522 nM T84133 CJV1G2 71455939 IC50 = 0.092 nM T84133 CVJ60C 71457356 IC50 = 0.22 nM T84133 CS54CU 71457642 Ki = 223 nM T84133 C1SWR4 71457643 Ki = 122 nM T84133 C8A9RD 71457644 Ki = 512 nM T84133 C8A4ME 71457746 IC50 = 0.075 nM T84133 CVY1U6 71459478 Ki = 4.5 nM T84133 CD3OM7 71459535 Ki = 93 nM T84133 COG41D 71459536 Ki = 98 nM T84133 C0YE2G 71459537 Ki = 422 nM T84133 C5HK3M 71459538 Ki = 121 nM T84133 C3VKH8 71459650 IC50 = 0.521 nM T84133 CHS8O5 71460995 Ki = 0.1 nM T84133 CH61LY 71461213 Ki = 3 nM T84133 CD3R9I 71461214 Ki = 8 nM T84133 C8B9OL 71461280 Ki = 7.9 nM T84133 CY9W5C 71461281 Ki = 843 nM T84133 CT6A8W 71461282 Ki = 991 nM T84133 CT2D6E 71461384 IC50 = 0.513 nM T84133 C73BXI 71462690 IC50 < 10 nM T84133 CS61KO 71520599 IC50 = 33 nM T84133 CT3IN6 71520691 IC50 = 33 nM T84133 C1D7QX 71520692 IC50 = 41 nM T84133 C1ADI4 71578082 IC50 < 100 nM T84133 C4GNJ3 71598545 IC50 > 1000 nM T84133 C9ASX2 71625031 IC50 = 991 nM T84133 CX7MY5 71680558 IC50 = 0.8 nM T84133 C68SDB 71719394 IC50 = 501.19 nM T84133 CU4RD3 71934591 IC50 = 530 nM T84133 CI6H0M 72163876 IC50 = 750 nM T84133 CMB3E6 72163877 IC50 = 660 nM T84133 CM57IJ 72163878 IC50 = 660 nM T84133 C8MIQ4 72163990 IC50 = 460 nM T84133 CUTR32 72163991 IC50 = 88 nM T84133 C7GO9N 72163992 IC50 = 87 nM T84133 CQV3Y9 72163993 IC50 = 24 nM T84133 CC2Q8Z 72164107 IC50 = 1600 nM T84133 CG9KC1 72164108 IC50 = 1600 nM T84133 CMH8P7 72164109 IC50 = 920 nM T84133 CP57OH 72164110 IC50 = 950 nM T84133 CZ0G2X 72165213 IC50 > 10000 nM T84133 C7XRY6 72190879 IC50 > 30000 nM T84133 COL24U 72193890 IC50 = 92 nM T84133 CKGQ16 72194628 IC50 = 0.15 nM T84133 CQ3GD7 72704434 Ki = 1800 nM T84133 CPIO30 72706193 IC50 > 10000 nM T84133 C1CQG9 72706253 IC50 = 1700 nM T84133 CF4W8Z 72706442 IC50 = 1600 nM T84133 C1H6MG 72724772 IC50 = 351.2 nM T84133 C98ESL 72724774 IC50 = 666.4 nM T84133 CPW50Y 72724856 IC50 = 4.85 nM T84133 C8O1UV 72724923 IC50 = 8.73 nM T84133 CWQ9G1 72724924 IC50 = 13.85 nM T84133 C9TQB6 72724925 IC50 = 0.9 nM T84133 CS4P2W 72724926 IC50 = 7.45 nM T84133 C2GUI0 72724927 IC50 = 18.48 nM T84133 C06ETS 72724928 IC50 = 5.12 nM T84133 CDOA38 72724979 IC50 = 6.88 nM T84133 CDTV07 72724982 IC50 = 157.1 nM T84133 CVC17O 72724984 IC50 = 6.73 nM T84133 CQ2S1U 72725040 IC50 = 8.96 nM T84133 CBM61I 73293715 IC50 = 403 nM T84133 CHR7D0 73334611 IC50 = 43 nM T84133 CQ9B4J 73387632 IC50 = 1590 nM T84133 CIE2C3 73387739 IC50 = 1790 nM T84133 C9ODB8 73387740 IC50 = 5 nM T84133 C5X6GJ 73387742 IC50 = 23 nM T84133 CT1E6V 73387743 IC50 = 21 nM T84133 C7D1SJ 73387744 IC50 = 83 nM T84133 CG89ET 73387745 IC50 = 25 nM T84133 CX65SQ 73387860 IC50 = 298 nM T84133 C3HSE2 73387863 IC50 = 171 nM T84133 CXOT45 73387957 IC50 = 1800 nM T84133 C74MPW 73387958 IC50 = 535 nM T84133 C3R0TC 73387959 IC50 = 11 nM T84133 CAL1N4 73387960 IC50 = 555 nM T84133 CHFG14 73425856 IC50 = 115 nM T84133 CEL2P4 73425857 IC50 = 639 nM T84133 C74TSX 73425972 IC50 = 87 nM T84133 CWX3M6 73425973 IC50 = 83 nM T84133 CEH2R6 73425974 IC50 = 20 nM T84133 CK5SA7 73425975 IC50 = 125 nM T84133 CPV3X9 73659152 Ki = 1100 nM T84133 C2FK6C 73659153 Ki = 5500 nM T84133 CVL07C 74049853 IC50 = 210 nM T84133 CT9Z7W 74049854 IC50 = 92 nM T84133 CA2R5W 74538674 IC50 < 100 nM T84133 C9JE6M 75815419 IC50 = 409 nM T84133 CSPU01 76210621 IC50 = 4.1 nM T84133 C16KIR 76283147 IC50 < 100 nM T84133 C8HPY6 76283633 IC50 = 200 nM T84133 C6ZO1T 76309994 IC50 > 1000 nM T84133 CVXP86 76309997 IC50 > 1000 nM T84133 C68NMU 76313712 IC50 > 1000 nM T84133 CGQ3L4 76313713 IC50 > 1000 nM T84133 CG4Y6I 76313715 IC50 = 309 nM T84133 CF91GV 76316930 Ki = 265 nM T84133 COR07S 76317224 IC50 = 849 nM T84133 CL03OP 76317226 IC50 > 1000 nM T84133 C8D5CS 76320933 IC50 > 1000 nM T84133 CKP16F 76320936 IC50 = 72 nM T84133 CQ8K4V 76320937 IC50 = 601 nM T84133 CNF60R 76320938 IC50 = 152 nM T84133 CTN90Q 76324596 IC50 = 16 nM T84133 CM9F4N 76324597 IC50 > 1000 nM T84133 C1WK7Z 76328150 IC50 = 99 nM T84133 C1YUL6 76328154 IC50 = 25 nM T84133 CCTF95 76328155 IC50 > 1000 nM T84133 CH0D1R 76328156 IC50 = 494 nM T84133 C41KHA 76328157 IC50 = 214 nM T84133 C2JPR1 76328158 IC50 = 166 nM T84133 CU2N9I 76328159 IC50 = 305 nM T84133 CFDQ21 76328160 IC50 = 180 nM T84133 C13ALF 76331835 IC50 = 299 nM T84133 CB76NH 76331836 IC50 = 774 nM T84133 CCY1F2 76331837 IC50 > 1000 nM T84133 CAV58P 76331838 IC50 = 89 nM T84133 CVC96N 76331839 IC50 = 208 nM T84133 C8CP3K 76903477 Ki = 0.23 nM T84133 CBTV14 77230235 Ki = 2200 nM T84133 CH90OK 80970089 Ki = 1200 nM T84133 CR95CP 80970101 Ki = 1000 nM T84133 C9E5LR 80970262 Ki = 220 nM T84133 CZ78LM 80970546 Ki = 890 nM T84133 CI43LO 80970589 Ki = 2100 nM T84133 C3NF5J 80970780 Ki = 880 nM T84133 CRE54Q 80970789 Ki = 2800 nM T84133 C3AFV8 80971037 Ki = 3600 nM T84133 CN8A4E 80971045 Ki = 1400 nM T84133 C1QLP8 80971247 Ki = 200 nM T84133 CET3Y9 80971319 Ki = 5300 nM T84133 CA92NJ 80971485 Ki = 1600 nM T84133 CX95WD 80971568 Ki = 130 nM T84133 CAUD50 80971601 Ki = 18 nM T84133 C9USK7 80971716 Ki = 51 nM T84133 C6RJP9 80972029 Ki = 6800 nM T84133 CYV42X 80972233 Ki = 37 nM T84133 CJ8S1R 80972289 Ki = 26 nM T84133 C5K6OY 80972640 Ki = 38 nM T84133 CK03GH 80978295 Ki = 4600 nM T84133 CQU45W 80978577 Ki = 1500 nM T84133 C9L8DC 81177397 Ki = 810 nM T84133 C50CVK 86291015 IC50 = 2.1 nM T84133 CV2GM7 86302601 IC50 = 24.2 nM T84133 C07WDK 86302602 IC50 = 41.5 nM T84133 CF1YH2 86302603 IC50 = 33.2 nM T84133 CM3R1U 86582302 IC50 = 20 nM T84133 C1P6DK 86582454 IC50 = 3 nM T84133 CTSL48 86688163 Ki = 12 nM T84133 C52BXE 86705377 IC50 > 10000 nM T84133 C6RB5X 86766620 Ki = 0.03 nM T84133 CTW8L6 86766622 Ki = 0.44 nM T84133 C9ZB8M 89586284 IC50 = 550 nM T84133 CZ4R0H 89586444 IC50 = 130 nM T84133 CP40LQ 89586661 IC50 = 1000 nM T84133 CZS95W 89586680 IC50 = 2400 nM T84133 CR4AW9 89593396 IC50 = 4.1 nM T84133 C1KY3L 89610300 IC50 = 0.12 nM T84133 CX9RL3 89621955 Ki = 8.5 nM T84133 CKHF70 89633452 Ki = 8.6 nM T84133 CN03MF 89763702 IC50 = 271 nM T84133 CUB2A8 90157072 Ki = 2.1 nM T84133 CF03DW 90168772 IC50 > 20000 nM T84133 CM6J9K 90168778 IC50 > 20000 nM T84133 C2BWK6 90644304 IC50 = 590 nM T84133 CG9H0I 90644305 IC50 = 6800 nM T84133 C17NSX 90644306 IC50 = 9.1 nM T84133 CC3YT0 90644307 IC50 = 8.3 nM T84133 CS3GT1 90644308 IC50 = 9.2 nM T84133 CELX01 90644309 IC50 = 28 nM T84133 CN01QJ 90644310 IC50 = 6.3 nM T84133 CTJ0H5 90644311 IC50 = 220 nM T84133 CF1IX2 90644312 IC50 = 37 nM T84133 CONS07 90644313 IC50 = 97 nM T84133 CW5HG6 90644314 IC50 = 200 nM T84133 CBMX19 90644315 IC50 = 7.3 nM T84133 C4XA2F 90644316 IC50 = 28 nM T84133 CMT94L 90644317 IC50 = 111 nM T84133 CGA67V 90644318 IC50 = 9.5 nM T84133 CCA0B1 90644319 IC50 = 1700 nM T84133 C3MRU1 90645023 IC50 = 15.1 nM T84133 CY9OX3 90645024 IC50 = 0.5 nM T84133 CWVQ98 90645025 IC50 = 5.7 nM T84133 CPZW52 90645026 IC50 = 115 nM T84133 C6GWH1 90645027 IC50 = 39.8 nM T84133 CU64KR 90645028 IC50 = 404 nM T84133 C7T4OL 90645029 IC50 = 105 nM T84133 C0A4ZG 90645030 IC50 = 36.8 nM T84133 C5J4ZG 90645031 IC50 = 51.5 nM T84133 CLQ9X5 90645032 IC50 = 21.5 nM T84133 C2DRU5 90645033 IC50 = 47.3 nM T84133 CO02RJ 90645034 IC50 = 20.7 nM T84133 CA2M6C 90645035 IC50 = 6.7 nM T84133 CX62CZ 90656262 IC50 = 123.2 nM T84133 CE7R3X 90656263 IC50 = 188.2 nM T84133 CPAX85 90656264 IC50 = 11.2 nM T84133 C01DHG 90656265 IC50 = 67.4 nM T84133 C6USP0 90656266 IC50 = 68.5 nM T84133 C3ONJ8 90656267 IC50 = 592.1 nM T84133 CQXK40 90656268 IC50 = 10.4 nM T84133 C5OGT4 90656269 IC50 = 5936.8 nM T84133 CVC4T3 90656270 IC50 = 3217.2 nM T84133 CZ6X5C 90656271 IC50 = 971.2 nM T84133 CNO3S8 90665367 IC50 = 610 nM T84133 C9MDB2 90665368 IC50 = 635 nM T84133 C1GUW7 90665369 IC50 = 3050 nM T84133 CE75WY 90665370 IC50 = 645 nM T84133 CR7ZV2 90665371 IC50 = 4250 nM T84133 C6IP3U 90665372 IC50 = 5150 nM T84133 CYU4G8 90665373 IC50 = 4600 nM T84133 CRJ8D4 90665374 IC50 = 0.4 nM T84133 C7F1IS 90665375 IC50 = 60 nM T84133 CZKD47 90665376 IC50 = 46 nM T84133 C0PWE2 90665377 IC50 = 168 nM T84133 CFB49U 90665378 IC50 = 415 nM T84133 C6NC2P 90665379 IC50 = 400 nM T84133 C2XOF1 90665380 IC50 = 635 nM T84133 C9F5QI 90668357 IC50 = 13900 nM T84133 CQR09V 90668358 IC50 = 7500 nM T84133 CXE08M 90668359 IC50 = 7400 nM T84133 C12BIU 90668360 IC50 = 10900 nM T84133 CG5HV8 90668361 IC50 = 0.24 nM T84133 C2HQ7I 90668362 IC50 = 0.36 nM T84133 C9VRW2 90668363 IC50 = 81.4 nM T84133 CDB74T 90668364 IC50 = 1.78 nM T84133 CTH48K 90668365 IC50 = 95 nM T84133 C07FTL 90668366 IC50 = 199 nM T84133 CX32TC 90668367 IC50 = 1850 nM T84133 C13GCO 90718236 IC50 = 6.3 nM T84133 C1JPD6 91844700 IC50 = 1.5 nM T84133 C60HAJ 91885643 Ki = 4.8 nM T84133 C7F6JY 92135987 IC50 = 27 nM T84133 CYQV05 92471958 IC50 = 510 nM T84133 CPO9J5 116378246 Ki = 680 nM T84133 CO3PG2 116386860 Ki = 1000 nM T84133 C4LER2 117728190 IC50 = 1.2 nM T84133 C1O7RV 117728381 IC50 = 4.4 nM T84133 C9TSE5 117728416 IC50 = 0.6 nM T84133 CH1P0N 117728473 IC50 = 7.4 nM T84133 CA46EP 117728534 IC50 = 3.2 nM T84133 C0G8NY 117728539 IC50 = 21.4 nM T84133 CWZ9R5 117728565 IC50 = 20.4 nM T84133 CIX1E9 117728795 IC50 = 2.2 nM T84133 CSCY01 117949009 IC50 > 10000 nM T84133 CYQ74R 118479645 IC50 = 1700 nM T84133 C0KPH4 118485600 IC50 > 10000 nM T84133 C43GZF 118485601 IC50 > 10000 nM T84133 C8UT1Z 118485623 IC50 > 10000 nM T84133 CC94IQ 118485651 IC50 = 59 nM T84133 CQ9X2T 118525749 IC50 = 35 nM T84133 CA9Z4N 118525753 IC50 = 96 nM T84133 COM19L 118525755 IC50 = 115 nM T84133 CCB0S9 118525772 IC50 = 67 nM T84133 C0SV3H 118525773 IC50 = 19.5 nM T84133 CG4Z8E 118525774 IC50 = 166 nM T84133 CQNY08 118525780 IC50 > 1000 nM T84133 CK3HY2 118525781 IC50 > 300 nM T84133 CGBK61 118525786 IC50 = 953 nM T84133 CYE6W5 118525795 IC50 = 135 nM T84133 C6IK4S 118525796 IC50 = 382 nM T84133 CE3UW6 118525799 IC50 = 172 nM T84133 C8OH0Y 118525801 IC50 = 146 nM T84133 CS23YQ 118525803 IC50 > 280 nM T84133 CP75JF 118525805 IC50 = 63 nM T84133 CCW37N 118525809 IC50 = 280 nM T84133 CR65SL 118525810 IC50 = 161 nM T84133 C5Y6KJ 118525812 IC50 > 1000 nM T84133 CVIU49 118525816 IC50 = 242 nM T84133 C94ZTQ 118525830 IC50 = 54 nM T84133 CM8IQ7 118525835 IC50 = 135 nM T84133 CF34RY 118525847 IC50 > 1000 nM T84133 CJX65U 118525848 IC50 = 280 nM T84133 CQ0LU1 118525854 IC50 = 52 nM T84133 C2PWK5 118534656 IC50 = 47 nM T84133 C5WDF6 118534657 IC50 = 794 nM T84133 C4H2LG 118534683 IC50 = 37 nM T84133 CR40SC 118534699 IC50 = 279 nM T84133 CVYK24 118556943 IC50 > 50000 nM T84133 CX0NV9 118658005 IC50 = 2.6 nM T84133 C01YKC 118658396 IC50 = 13 nM T84133 CSKE85 118707952 IC50 = 20.9 nM T84133 CZY9E8 118707953 IC50 = 115.7 nM T84133 C52ELD 118707954 IC50 = 102.6 nM T84133 C8WQO0 118707955 IC50 = 18.2 nM T84133 CNF3J2 118707956 IC50 = 29.2 nM T84133 CB2C3R 118707957 IC50 = 266.7 nM T84133 CO20GE 118707958 IC50 = 177.2 nM T84133 CZR3G0 118707959 IC50 = 153.1 nM T84133 CBRP26 118707960 IC50 = 8.54 nM T84133 CD67FM 118707961 IC50 = 19.1 nM T84133 C5VPF6 118707962 IC50 = 128.1 nM T84133 CZ31HQ 118707963 IC50 = 71 nM T84133 CJ0G3M 118707964 IC50 = 1.3 nM T84133 C1YX7I 118707965 IC50 = 0.3 nM T84133 C6G7DB 118707966 IC50 = 2.6 nM T84133 C0RCP5 118707967 IC50 = 135.5 nM T84133 CC5X3L 118707968 IC50 = 552.1 nM T84133 CD65SB 118708350 IC50 = 40 nM T84133 COV3E5 118708351 IC50 = 170 nM T84133 CTF9R5 118708352 IC50 = 220 nM T84133 CF7NI4 118708353 IC50 = 1300 nM T84133 CW74UJ 118708354 IC50 = 190 nM T84133 CI1Y9A 118708355 IC50 = 42 nM T84133 C9HR7F 118708356 IC50 = 40 nM T84133 CI18GD 118708357 IC50 = 55 nM T84133 CF68VD 118708358 IC50 = 480 nM T84133 CQ52CE 118708359 IC50 = 900 nM T84133 CMX51I 118708360 IC50 = 1000 nM T84133 C4I9AY 118721431 IC50 = 21000 nM T84133 CIQ2R0 118721671 IC50 = 1000 nM T84133 CY0LR7 118725353 IC50 = 18.4 nM T84133 CBAF10 118725354 IC50 = 4250 nM T84133 C5F3PM 118725355 IC50 = 14 nM T84133 C31ARB 118725356 IC50 = 1550 nM T84133 C5TL8H 118725359 IC50 = 2.86 nM T84133 C7EYI4 118725362 IC50 = 9.8 nM T84133 C5VTG0 118725363 IC50 = 350 nM T84133 C54GSD 118725364 IC50 = 518 nM T84133 C70GAC 118725365 IC50 = 79.3 nM T84133 CP9L2X 118725366 IC50 = 18.6 nM T84133 CEI6R3 118725367 IC50 = 8 nM T84133 CE49ML 118725368 IC50 = 3.73 nM T84133 C1AG7N 118725371 IC50 > 1900 nM T84133 CVDC45 121596889 IC50 = 2.4 nM T84133 C96LCR 122182051 IC50 = 1800 nM T84133 C2WP3Y 122182052 IC50 = 64 nM T84133 CZ2P0D 122182053 IC50 = 330 nM T84133 CXWB12 122185004 IC50 = 3 nM T84133 C8HFW5 122185005 IC50 = 1 nM T84133 CRJE23 122185011 IC50 = 252 nM T84133 C9T3ER 122191265 Ki = 180 nM T84133 CS5UJ1 122192111 Ki = 540 nM T84133 C4QPE7 122192112 Ki = 1300 nM T84133 C5VQJ7 122192113 Ki = 10 nM T84133 C8DIW9 122192114 Ki = 5.1 nM T84133 CMS3N6 122192115 Ki = 590 nM T84133 CS54NV 122192116 Ki = 400 nM T84133 CC3DO7 122192117 Ki = 0.047 nM T84133 CQDZ58 122192118 Ki = 0.055 nM T84133 CS6D4W 122192119 Ki = 0.11 nM T84133 C5XBU8 122192120 Ki = 0.37 nM T84133 CS70BK 122192925 Ki = 87 nM T84133 CI87VG 122192926 Ki = 280 nM T84133 COM57X 122192927 Ki = 123 nM T84133 C6Z1LU 122192928 Ki = 265 nM T84133 C41RCJ 122192929 Ki = 49 nM T84133 CM6ZQ8 122192930 Ki = 61 nM T84133 CV3MK1 122192931 Ki = 64 nM T84133 CJRB26 122192932 Ki = 171 nM T84133 C57BRI 122192933 Ki = 163 nM T84133 CW2O7J 122192934 Ki = 45 nM T84133 C5D4VJ 122192935 Ki > 1000 nM T84133 CEI01K 122192936 Ki = 39 nM T84133 CP3AS6 122192937 Ki = 15 nM T84133 C6ZHK9 122192938 Ki = 13 nM T84133 CIH0P5 122192939 Ki = 7.7 nM T84133 C20PAT 122192940 Ki = 30 nM T84133 CQD1I9 122192941 Ki = 6.3 nM T84133 CVGX87 122192953 Ki = 1 nM T84133 C0DNH8 122192954 Ki = 1.8 nM T84133 CAIJ87 122192955 Ki = 0.025 nM T84133 CN98GL 122193004 Ki = 1124 nM T84133 C1PKY7 122193005 Ki = 109 nM T84133 CS6M9C 122193679 IC50 > 100000 nM T84133 CJKO62 122193703 IC50 = 0.71 nM T84133 C9W1JO 122193704 IC50 = 0.68 nM T84133 C2MNX0 122193705 IC50 = 1.8 nM T84133 C5EHB7 122193706 IC50 = 0.32 nM T84133 C5WI6U 122193707 IC50 = 0.65 nM T84133 COT0R6 122193708 IC50 = 0.27 nM T84133 CJF36H 122193709 IC50 = 0.24 nM T84133 C0J6MS 122193710 IC50 = 0.33 nM T84133 C0XLR7 122193711 IC50 = 0.52 nM T84133 CC9I0U 122193712 IC50 = 3.07 nM T84133 CX30HD 122193713 IC50 = 0.26 nM T84133 CU5O4D 122193714 IC50 > 76 nM T84133 C07INS 122193715 IC50 = 33.5 nM T84133 C6IJH8 122193928 IC50 = 1.16 nM T84133 CNT17O 122193929 IC50 = 1.12 nM T84133 C6Q5UO 122193930 IC50 = 0.36 nM T84133 C1SWM0 122193931 IC50 = 0.47 nM T84133 C9JSX0 122193932 IC50 = 0.3 nM T84133 C6GI3B 122193933 IC50 = 0.37 nM T84133 C9PTW4 122193934 IC50 = 4.98 nM T84133 C5FKM8 122193935 IC50 = 0.76 nM T84133 C4IH7Q 122194381 IC50 = 0.23 nM T84133 CV07GU 122196327 IC50 = 2435.5 nM T84133 CT53EP 122196328 IC50 = 2740.1 nM T84133 C1MO9A 122196329 IC50 = 364.2 nM T84133 CU4N9V 122196331 IC50 = 350.9 nM T84133 CC6SY1 122196335 IC50 = 120.1 nM T84133 CUFV13 122196338 IC50 = 226.6 nM T84133 C3W6MK 122196339 IC50 = 193.6 nM T84133 C31DAM 122196340 IC50 = 1.12 nM T84133 C8K9XA 122196341 IC50 = 1.62 nM T84133 CK2A0O 122196342 IC50 = 1.11 nM T84133 C3CKT2 122196343 IC50 = 2.71 nM T84133 CPD5U0 122196344 IC50 = 1.23 nM T84133 CDWR01 122196345 IC50 = 1.41 nM T84133 CPNO72 122196346 IC50 = 5.02 nM T84133 CBHJ25 122196347 IC50 = 1.85 nM T84133 CFR30U 122196348 IC50 = 6.46 nM T84133 CE9N4M 122196392 IC50 = 1.9 nM T84133 CNA5E2 122196393 IC50 = 18.62 nM T84133 CC46NG 122196394 IC50 = 1.22 nM T84133 CCV89J 122196396 IC50 = 21.2 nM T84133 C2ZV9X 122196397 IC50 = 21.69 nM T84133 C9OG6C 122196398 IC50 = 136.6 nM T84133 CP27SM 122196399 IC50 = 926.4 nM T84133 CBN5D2 122196400 IC50 = 0.21 nM T84133 C2FMR4 122196401 IC50 = 0.33 nM T84133 CR19NH 122196402 IC50 = 0.3 nM T84133 C9I0FA 122196403 IC50 = 0.54 nM T84133 C5P8EK 122196404 IC50 = 1.73 nM T84133 C9AEK1 122196405 IC50 = 0.73 nM T84133 C8WYE5 122196406 IC50 = 11.96 nM T84133 C0M3DA 122196407 IC50 > 10000 nM T84133 C5WBC8 122196408 IC50 = 2984.5 nM T84133 CM3D6N 122196409 IC50 = 28.9 nM T84133 C2RMU9 122196410 IC50 = 41.5 nM T84133 C10LCF 122196411 IC50 = 37 nM T84133 C48VJC 122196412 IC50 = 3.3 nM T84133 CVX7U9 127029185 IC50 > 20000 nM T84133 C4UR7D 127038167 IC50 = 2.95 nM T84133 C4H2TJ 127038168 IC50 = 3.3 nM T84133 CL9JT8 127038169 IC50 = 0.12 nM T84133 CN9BH4 127038170 IC50 = 0.048 nM T84133 CC0L8Y 127038242 Ki = 8.3 nM T84133 CO2CI9 127038507 IC50 = 3.18 nM T84133 CRF5C6 127038508 IC50 = 1.57 nM T84133 CJPX60 127038509 IC50 = 0.11 nM T84133 C7X2VQ 127038510 IC50 = 26.3 nM T84133 C26EAG 127038511 IC50 = 0.41 nM T84133 CTM9E4 127038512 IC50 = 0.33 nM T84133 C6AQ2U 127038513 IC50 = 0.99 nM T84133 CJ1Z4H 127038575 Ki = 1.4 nM T84133 C6HZ8P 127038725 IC50 = 10.3 nM T84133 CV1FM0 127038868 IC50 = 0.87 nM T84133 CADU23 127038869 IC50 = 0.037 nM T84133 C50MRW 127040517 IC50 = 0.46 nM T84133 CAG7Y1 127040518 IC50 = 20.4 nM T84133 CLY63Q 127040519 IC50 = 1.69 nM T84133 C0RT1M 127040594 Ki = 3.1 nM T84133 C95LEY 127041240 IC50 = 110 nM T84133 C8NLE7 127041841 Ki = 0.006 nM T84133 C7VM1D 127041864 Ki = 1.1 nM T84133 CM7Y0H 127041887 Ki = 0.01 nM T84133 CMP85X 127041888 Ki = 0.02 nM T84133 COM5Q1 127042152 Ki = 0.02 nM T84133 C0Q6TF 127042166 Ki = 3.1 nM T84133 CNWS83 127042167 Ki = 19.1 nM T84133 CK7X3P 127042168 Ki = 4.1 nM T84133 CRL5T7 127042169 Ki = 0.4 nM T84133 CC78KF 127042170 Ki = 1.1 nM T84133 CB74PN 127042524 Ki = 15.5 nM T84133 C42NGM 127042525 Ki = 1.7 nM T84133 C9G8FY 127042526 Ki = 0.01 nM T84133 CW38DL 127042532 IC50 = 16 nM T84133 CH9PI1 127042533 IC50 = 120 nM T84133 C8GS0B 127042534 IC50 = 490 nM T84133 CC3W0Z 127042551 Ki = 20.3 nM T84133 C1QGB8 127042552 Ki = 3.6 nM T84133 C4D1OU 127042553 Ki = 54 nM T84133 CVX07H 127042560 Ki = 58 nM T84133 CXK9V3 127049326 IC50 = 2800 nM T84133 CG26VL 127049327 IC50 = 25 nM T84133 CPIX38 127049328 IC50 = 760 nM T84133 C2LGT3 129051755 IC50 = 458 nM T84133 C62CSI 129051756 IC50 = 69 nM T84133 C5RFV2 129051760 IC50 = 84 nM T84133 CH20AQ 129051764 IC50 = 40 nM T84133 CDJ2V1 129051781 IC50 = 198 nM T84133 CUE8J7 129051785 IC50 = 268 nM T84133 C7AD3Z 129051788 IC50 = 28 nM T84133 CACJ46 132489333 IC50 = 153 nM T84133 C9GNP7 132502926 IC50 = 38 nM T84133 CTH6R5 132538329 IC50 = 2 nM T84133 C2P1IU 134129996 IC50 > 100000 nM T84133 CLE03O 134130328 IC50 > 100000 nM T84133 CSN6J0 134130563 IC50 > 100000 nM T84133 C0A1CZ 134131162 IC50 > 100000 nM T84133 C5FTY2 135400457 Ki = 990000 nM T84133 CTR37Z 135408753 Ki = 910000 nM T84133 CB8YM4 135408756 Ki = 450000 nM T84133 CHDC83 135566745 IC50 > 10000 nM T84133 C9IJK1 135566935 IC50 = 6900 nM T84133 CMWA73 136042357 IC50 = 1720 nM T84133 CRP24A 136087045 IC50 = 33300 nM T84133 C7SUX4 136087050 IC50 = 3700 nM T84133 C8UF7G 136087052 IC50 > 50000 nM T84133 CGI17Y 136147441 IC50 < 500 nM T84133 C21FVA 136180322 IC50 = 2000 nM T84133 CQW7T0 136197286 IC50 > 10000 nM T84133 C8TQ7A 136217455 IC50 > 50000 nM T84133 CN8PK6 136927883 IC50 = 8.5 nM T84133 C08KZR 137007094 IC50 = 10800 nM T84133 CQK3V2 137007095 IC50 = 6620 nM T84133 CLE62X 137179301 IC50 = 117 nM T84133 C8FD1X 137243493 IC50 = 3800 nM T84133 CUM3T5 137243503 IC50 > 30000 nM T84133 C9IK5Q 137243508 IC50 = 280 nM T84133 C1JUS2 137243509 IC50 = 100 nM T84133 CI1J9K 137289913 IC50 = 3.3 nM T84133 C74KSG 137332065 IC50 = 1.7 nM T84133 C2N9VT 137348687 IC50 = 7400 nM T84133 CE1MA9 137631455 IC50 = 62 nM T84133 C0YMI5 137631826 IC50 > 10000 nM T84133 C5TDQ8 137632065 IC50 = 61 nM T84133 CQFK31 137633676 IC50 = 243 nM T84133 CGC75I 137633691 IC50 = 68 nM T84133 CAM92S 137634864 IC50 = 391 nM T84133 CIMX51 137636423 IC50 = 75 nM T84133 CAGV95 137636529 IC50 = 327 nM T84133 CX23JH 137637969 IC50 = 60 nM T84133 C1WAT7 137640957 IC50 = 130 nM T84133 CXWU26 137641682 IC50 = 107 nM T84133 C90CHG 137642556 IC50 = 168 nM T84133 C2XW5T 137643774 IC50 = 103 nM T84133 CQC5R0 137644374 IC50 = 116 nM T84133 C1Y7TO 137644422 IC50 = 447 nM T84133 C7MAO1 137645978 IC50 = 113 nM T84133 C24PNB 137650825 IC50 = 336 nM T84133 C2HS7D 137651999 IC50 = 56 nM T84133 C5XH7C 137653888 IC50 = 529 nM T84133 C6C7XH 137655649 IC50 = 452 nM T84133 C7LPA8 137655726 IC50 = 119 nM T84133 CP7Q5D 137656637 IC50 = 76 nM T84133 C7OH1C 137658687 IC50 = 518 nM T84133 CRD93N 137659470 IC50 = 168 nM T84133 CKEY52 137660104 IC50 = 258 nM T84133 C6KYD7 137700754 IC50 = 7310 nM T84133 CM3UF7 137700779 IC50 = 0.44 nM T84133 CPTE92 138319693 IC50 = 46 nM T84133 C2QLX3 138393292 IC50 = 920 nM T84133 CF6B8H 138857395 IC50 = 294 nM T84133 C72GWA 138857396 IC50 = 2.9 nM T84133 C7AHV4 138857397 IC50 = 28 nM T84133 CMW20N 141737696 IC50 > 4000 nM T84133 C8HEG7 141737705 IC50 > 3000 nM T84133 CC64PE 145949747 IC50 = 884 nM T84133 CU9YW0 145950008 IC50 = 381 nM T84133 C0F5PO 145950382 IC50 > 1000 nM T84133 C7Z5JP 145952479 IC50 = 280 nM T84133 CNIV78 145952823 IC50 = 770 nM T84133 C70YLA 145953136 IC50 = 76 nM T84133 C0C6FG 145954733 IC50 = 107 nM T84133 CQN9P3 145954872 IC50 = 163 nM T84133 C2KN1T 145955431 IC50 > 5000 nM T84133 C36IDE 145957514 IC50 > 1000 nM T84133 CW0JY3 145957704 IC50 > 1000 nM T84133 CH7VB3 145957961 IC50 = 145 nM T84133 CMTR43 145958975 IC50 = 268 nM T84133 CYZR45 145959927 IC50 = 315 nM T84133 C37PRT 145967337 IC50 < 100 nM T84133 CF25ZG 145967398 IC50 = 100 nM T84133 CAR1K5 145972948 IC50 = 581 nM T84133 CC7HN2 145974174 IC50 > 100000 nM T84133 CD5P0M 145974821 IC50 > 280 nM T84133 CK1BR0 145978345 IC50 > 100000 nM T84133 CHJ79V 145997874 IC50 > 10000 nM T84133 CY1R9G 147132320 IC50 = 403 nM T84133 C2AHD9 148588374 IC50 = 0.87 nM T84133 CD38ZO 155513157 IC50 = 44 nM T84133 C83XTD 155514176 IC50 = 5.2 nM T84133 C48WQL 155514804 IC50 = 441 nM T84133 C14BPA 155515110 IC50 = 2083 nM T84133 CQAY86 155517940 IC50 = 0.3 nM T84133 C49UIO 155519155 IC50 = 20 nM T84133 CE2MO6 155519440 IC50 = 47 nM T84133 CZM1V6 155520000 IC50 = 138 nM T84133 CF4B7U 155520076 IC50 = 75 nM T84133 CT7K4A 155520403 IC50 = 69 nM T84133 CI6AT8 155520893 IC50 = 44 nM T84133 CUA1X6 155521116 IC50 = 287 nM T84133 CL8CU6 155521936 IC50 > 200000 nM T84133 CWS0T8 155522940 IC50 = 510 nM T84133 CPZ9C5 155523000 IC50 = 1219 nM T84133 CPIE52 155524256 IC50 = 1476 nM T84133 C4J8EY 155524365 IC50 = 0.061 nM T84133 CGY0B7 155526339 IC50 = 292 nM T84133 CX7D8K 155526808 IC50 > 10000 nM T84133 CMPE29 155527485 IC50 = 8.4 nM T84133 C7ERC3 155527562 IC50 = 1 nM T84133 C4PE7I 155528020 IC50 = 78 nM T84133 C47UVA 155528950 IC50 = 105 nM T84133 CVG71O 155529178 IC50 = 105 nM T84133 CQPC31 155530033 IC50 = 110 nM T84133 C74GVU 155530078 IC50 = 279 nM T84133 CZAP29 155530397 IC50 = 416 nM T84133 CT85RG 155530589 IC50 > 200000 nM T84133 CUS48O 155530649 IC50 = 23 nM T84133 C73WIM 155530814 IC50 = 74 nM T84133 C7SI1U 155531139 IC50 = 320 nM T84133 CICH53 155532871 IC50 = 135 nM T84133 C6POE9 155533544 IC50 = 52 nM T84133 C3ZE6S 155535535 IC50 = 12 nM T84133 C8J0FO 155535672 IC50 = 23 nM T84133 CRA93Z 155539143 IC50 = 182 nM T84133 C84NIR 155540213 IC50 = 13.8 nM T84133 C6KEO7 155542008 IC50 = 88 nM T84133 C5QCM6 155545348 IC50 = 4.7 nM T84133 CAK63Q 155545457 IC50 = 0.76 nM T84133 CAD3C9 155545902 IC50 = 123 nM T84133 C7PQ5B 155546577 IC50 = 200 nM T84133 CAD6U2 155546988 IC50 = 2.1 nM T84133 CO3W9J 155549412 IC50 = 23 nM T84133 CXK67C 155551574 IC50 = 440 nM T84133 CZV45E 155554965 IC50 = 275 nM T84133 C2OYG0 155555420 IC50 = 10 nM T84133 CP18OF 155555969 IC50 > 1000 nM T84133 CJE59L 155558096 IC50 = 120 nM T84133 C2DA1W 155561694 IC50 > 500000 nM T84133 CC8I1S 155566153 IC50 = 1920 nM T84133 C95JGC 155566500 IC50 = 62 nM T84133 CT2SY1 155568004 IC50 = 7.6 nM T84133 CQ2R0W 155568588 IC50 > 500000 nM T84133 CYAZ51 66678448 Ki = 0.95 nM T84133 CF8Z7Y 69932178 IC50 = 0.06 nM T84133 D06NIT 135564899 IC50 > 1000 nM T84133 D09RKU 46239428 Ki = 5 nM T84133 D0V4WB 149790 IC50 > 16000 nM T84133 D0VB2W 21501 Ki = 560000 nM T65019 D00MDP 466151 IC50 = 0.3 nM T65019 D0Q8CS 60937 IC50 = 30500 nM T65019 D0VM2L 68740 IC50 = 12600 nM T65019 D05VZE 119031 IC50 = 1.82 nM T65019 D0A4RF 657061 IC50 = 22.91 nM T65019 D0MW3H 9824350 IC50 = 23 nM T65019 D0U2BH 65064 IC50 = 6800 nM T65019 D0G1LL 74221072 IC50 = 50000 nM T65019 D0N6ZA 74221131 IC50 > 100000 nM T65019 D0UM5R 74221070 IC50 = 15000 nM T65019 D01DVX 9847838 IC50 = 499 nM T65019 D03BOZ 3342298 IC50 = 1.1 nM T65019 D0E5GY 9904965 IC50 = 1.9 nM T65019 D0N8NK 11641563 IC50 = 2220 nM T65019 D0P8YC 5362422 IC50 = 2.9 nM T65019 D0T9HG 132519 IC50 = 0.41 nM T65019 C4U7SY 401129 IC50 = 12500 nM T65019 C4D7TS 448002 IC50 = 13 nM T65019 CC54LQ 450256 IC50 > 100000 nM T65019 CG1I8P 467296 IC50 = 15600 nM T65019 CTPW02 467297 IC50 = 3700 nM T65019 CS4O7K 685005 IC50 > 500000 nM T65019 CP1Q6R 703233 IC50 = 55000 nM T65019 C9IFC6 1348435 IC50 = 21000 nM T65019 CN9C8D 2140735 IC50 = 310000 nM T65019 CN6E3U 2366268 IC50 = 7500 nM T65019 CY3TD6 3348132 Ki = 105 nM T65019 C3EI6T 4085085 IC50 = 51000 nM T65019 CBN96T 4358655 IC50 > 100000 nM T65019 CC5O4E 4369384 IC50 = 6500 nM T65019 CZS0G5 5276565 IC50 > 100000 nM T65019 C3JN0F 5277465 IC50 = 33500 nM T65019 CRJK67 5277481 IC50 > 100000 nM T65019 CYF7S5 5277490 IC50 > 100000 nM T65019 CP7BG0 6852146 IC50 = 2200 nM T65019 CN5L2B 6852147 IC50 = 79 nM T65019 CP2XK7 6882342 IC50 = 150000 nM T65019 C76RCQ 9801569 IC50 = 963 nM T65019 CIXD67 9802768 IC50 = 8 nM T65019 CQ46XD 9804842 IC50 = 1700 nM T65019 CTK6J8 9808181 IC50 = 66900 nM T65019 C9RQM7 9808674 IC50 = 7.4 nM T65019 C6KJ9W 9822461 IC50 = 47 nM T65019 C6IX7G 9822926 IC50 = 5.6 nM T65019 CE9AL3 9847113 IC50 = 10.6 nM T65019 C4IEK0 9850035 IC50 = 108 nM T65019 CI8Z0R 9866250 IC50 = 7.4 nM T65019 CJS23I 9868333 Ki > 5290 nM T65019 CLQ29X 9869597 IC50 = 1710 nM T65019 CHU9I8 9871883 IC50 = 4.6 nM T65019 C0ZT7A 9883002 Ki = 37 nM T65019 C3ZG6O 9887870 IC50 = 240 nM T65019 CD79UJ 9890632 IC50 > 100000 nM T65019 CH69LT 9892815 IC50 = 13 nM T65019 CSIB97 9896504 IC50 > 100000 nM T65019 C4YGT6 9928325 IC50 = 56 nM T65019 C03GVA 9932290 Ki = 240 nM T65019 CDXR37 9933197 IC50 = 64 nM T65019 C65ION 9935032 IC50 = 500 nM T65019 CG38KL 9936728 Ki = 140 nM T65019 CQY54S 9952396 IC50 = 88 nM T65019 C9X0YR 9954867 IC50 > 10000 nM T65019 C3Q2UJ 9956686 IC50 = 200 nM T65019 CI5TW9 9956699 IC50 = 20100 nM T65019 CC4WG3 9957228 Ki > 300000 nM T65019 CN76XI 9957653 IC50 = 7 nM T65019 C9DRB7 9966028 IC50 = 2900 nM T65019 CUA65C 9982414 IC50 = 150 nM T65019 CR7T3J 10009978 Ki > 2000 nM T65019 CW2MK1 10043732 Ki = 210 nM T65019 C7O8HD 10044261 IC50 = 2.5 nM T65019 C7CT4E 10045150 IC50 = 1.9 nM T65019 CCF5Z4 10047585 IC50 = 2.08 nM T65019 CB9S7N 10101618 IC50 = 19 ug.mL-1 T65019 C0G7IY 10114318 Ki = 200 nM T65019 CVK61T 10116047 IC50 = 11 nM T65019 C78JHL 10116107 Ki = 390 nM T65019 C7A8MI 10120093 IC50 = 3.7 nM T65019 C7KR3Y 10136680 Ki = 150 nM T65019 CNU93J 10136924 Ki = 440 nM T65019 C1CDF2 10136925 Ki = 330 nM T65019 CJ9EX4 10138303 Ki = 250 nM T65019 CO6PS3 10162900 Ki = 180 nM T65019 CR5H6E 10163627 Ki > 5290 nM T65019 CCX3T6 10183064 Ki = 3070 nM T65019 CK0P3F 10186536 Ki > 5290 nM T65019 CE1LI3 10204303 Ki = 180 nM T65019 CQFP69 10206106 Ki = 340 nM T65019 C4K1MJ 10208262 Ki > 5290 nM T65019 CV5X8A 10224181 IC50 > 30000 nM T65019 CGKU70 10224396 Ki = 240 nM T65019 C2MES9 10271604 Ki > 100000 nM T65019 CGP97S 10274748 Ki = 100 nM T65019 C3IG0K 10280852 IC50 = 4.1 nM T65019 CDU36Y 10296475 Ki = 590 nM T65019 C48IRP 10296785 Ki = 50 nM T65019 CY08WJ 10322755 Ki = 163 nM T65019 C7UZA4 10340758 IC50 = 8.5 nM T65019 C6WZ4F 10367355 IC50 = 34 nM T65019 CFKA79 10395015 Ki = 2000 nM T65019 C5WV1N 10439082 Ki > 2000 nM T65019 C8M9FE 10462640 Ki = 160000 nM T65019 CNQZ36 10483139 Ki > 10000 nM T65019 C9C5EL 10521197 IC50 = 2.3 nM T65019 C21VZS 10573362 IC50 = 17.6 nM T65019 C3R2SO 10580533 Ki = 105 nM T65019 C6FWC1 10808125 IC50 = 13 nM T65019 C2A0IX 10833840 IC50 = 105 nM T65019 C9WPH7 11016072 Ki = 740 nM T65019 CBE68H 11016073 Ki = 330 nM T65019 CR4V2D 11101785 Ki = 380 nM T65019 CD1Q0L 11157488 IC50 = 20000 nM T65019 CEL1F0 11248884 IC50 = 5600 nM T65019 CO7T3M 11261246 IC50 = 7.7 nM T65019 CP17ID 11284983 IC50 = 15000 nM T65019 C1IW7N 11292680 IC50 = 9.8 nM T65019 C8C5AV 11294179 Ki > 10000 nM T65019 CLH50U 11318841 IC50 = 15800 nM T65019 CJ5SU9 11328354 Ki > 300000 nM T65019 C0XR3B 11330861 IC50 = 50118.72 nM T65019 CQH57S 11342435 IC50 = 5000 nM T65019 CU04HF 11419551 IC50 = 13900 nM T65019 COS67B 11456566 IC50 = 30000 nM T65019 C96DRO 11466734 IC50 = 5450 nM T65019 C7QF0G 11467517 IC50 = 11200 nM T65019 CWS35C 11510523 IC50 = 20700 nM T65019 C5VUM2 11517085 Ki = 140 nM T65019 CQ9E6J 11519157 IC50 = 4735 nM T65019 C5MO0U 11526826 IC50 = 1641 nM T65019 C9Y6LH 11533683 IC50 = 19700 nM T65019 CCW1B8 11569185 IC50 = 3121 nM T65019 CW5A4S 11569716 IC50 = 1305 nM T65019 CHV2G1 11575995 Ki > 10000000 nM T65019 CL9K7T 11583525 IC50 = 1950 nM T65019 CTQ87G 11599024 IC50 = 13000 nM T65019 C8IWM1 11605689 IC50 = 553 nM T65019 C0VCJ8 11613810 IC50 = 220 nM T65019 CCBS59 11634234 IC50 = 3642 nM T65019 CNY92D 11640694 Ki > 40000 nM T65019 C1U3EX 11656290 IC50 > 10000 nM T65019 C28WNK 11682752 Ki = 900 nM T65019 CRF7V9 11691964 IC50 = 915 nM T65019 C3U6ZR 11697504 Ki = 11000 nM T65019 C2BJ3X 11716217 Ki = 31910 nM T65019 CCD93H 11730086 Ki = 110 nM T65019 CO8QT0 11753905 Ki = 2800 nM T65019 C4XR5G 11963536 IC50 = 24000 nM T65019 C02BWA 11967143 Ki > 2000 nM T65019 CB80OT 12000718 IC50 > 20000 nM T65019 C43PJZ 12000720 IC50 > 20000 nM T65019 C0K8ZX 12404978 IC50 > 500000 nM T65019 CQTX49 13738810 IC50 > 100000 nM T65019 C8TH1O 14177156 IC50 > 500000 nM T65019 C3N1KV 15629940 IC50 > 100000 nM T65019 CB3A4Z 15941413 Ki = 215 nM T65019 CA40FE 15941550 Ki = 90 nM T65019 CM3D1L 15941553 Ki = 680 nM T65019 CQ0ZL7 15941677 Ki = 145 nM T65019 C6F9WV 15941679 Ki = 360 nM T65019 C7C1HI 15941680 Ki = 240 nM T65019 C6R1LD 15985818 IC50 = 582 nM T65019 CL7KX3 16040152 IC50 = 0.57 ug.mL-1 T65019 CTZ3R1 16040153 IC50 = 3.2 ug.mL-1 T65019 CS46XU 16126723 IC50 = 14 nM T65019 C91EXN 16655061 IC50 = 14800 nM T65019 CQS0F5 16719301 IC50 > 10000 nM T65019 C75XDI 16730519 IC50 > 5000 nM T65019 C50AEZ 18616892 IC50 > 10000 nM T65019 CIEH93 19382975 IC50 = 69000 nM T65019 CK8MP3 20620240 Ki > 10000 nM T65019 CPC4G6 20620273 Ki > 10000 nM T65019 C2E3CY 20620614 Ki > 10000 nM T65019 CC7BF2 20636126 IC50 = 616.6 nM T65019 C6A1QE 20636128 IC50 = 645.65 nM T65019 C4JPZ3 20636129 IC50 = 9332.54 nM T65019 CAU28R 20636149 IC50 = 8709.64 nM T65019 CXS53V 20636183 IC50 = 36.31 nM T65019 C18RXS 20735191 IC50 = 9.5 nM T65019 C4I1OM 20735209 IC50 = 10000 nM T65019 CIC4S9 22004232 IC50 = 71 nM T65019 CZT05X 22484417 Ki > 10000 nM T65019 CZT64B 22484431 Ki > 10000 nM T65019 CAM10T 22485252 IC50 = 24 nM T65019 CBJS34 22485260 IC50 = 3.63 nM T65019 C9MU7N 22485263 IC50 > 10000 nM T65019 CEGJ03 22485276 IC50 = 3486 nM T65019 C7VB8G 22485289 IC50 = 0.73 nM T65019 CNB02I 22485291 IC50 = 10.5 nM T65019 CAY3N6 22485292 IC50 = 159 nM T65019 C94OCJ 22485302 IC50 = 6.8 nM T65019 C3YL5X 22485311 IC50 = 53.9 nM T65019 CWA03L 22485327 IC50 = 3.1 nM T65019 C6JRW5 22485340 IC50 = 13.3 nM T65019 C5JZF1 22485344 IC50 = 47 nM T65019 CI7MY5 22485346 IC50 = 20 nM T65019 CI1YL7 22485347 IC50 = 4 nM T65019 C25OBD 22485356 IC50 = 4.5 nM T65019 C7I0EW 22485367 IC50 = 1.71 nM T65019 CL64TJ 22485368 IC50 = 100.5 nM T65019 CT4GF9 22485381 IC50 > 10000 nM T65019 C27NDB 22485386 IC50 = 160 nM T65019 CTJ9I3 22485392 IC50 = 25.8 nM T65019 C3MG9P 22485396 IC50 = 83 nM T65019 CZY10U 22485408 IC50 = 58.6 nM T65019 C89AGT 22485413 IC50 = 14.9 nM T65019 C8GHU9 22485432 IC50 = 49.4 nM T65019 C9BT5F 22626996 IC50 = 784 nM T65019 C2Q4XK 22707806 IC50 = 9 nM T65019 CIYA45 22985930 IC50 = 53.3 nM T65019 CX32YK 23513795 IC50 = 257 nM T65019 C6IZ1S 23513821 IC50 = 2080 nM T65019 CPNM93 23513825 IC50 = 489 nM T65019 CML90Q 23513831 IC50 = 889 nM T65019 C4R2AJ 23625454 IC50 = 4891 nM T65019 C4R2DA 23645953 Ki > 300000 nM T65019 CWN3I4 23645959 Ki > 300000 nM T65019 CL24JR 23655078 IC50 = 3290 nM T65019 CBI81H 23672150 IC50 = 15 ug.mL-1 T65019 C7KF1N 23729138 IC50 = 2000 nM T65019 CG3J2L 24768528 IC50 = 2370 nM T65019 C5M3YW 24799779 Ki = 2400000 nM T65019 CE29HI 24860424 IC50 = 4320 nM T65019 CT10JE 24860425 IC50 = 3619 nM T65019 CRC98J 24860426 IC50 = 1000 nM T65019 C8MKR0 24860427 IC50 = 7047 nM T65019 CNR3U7 24866945 IC50 = 20000 nM T65019 C4UEM5 24871537 Ki > 50000 nM T65019 CP2L5B 24871655 Ki > 50000 nM T65019 C4SP3O 24936157 IC50 = 3.9 nM T65019 CAQ9Z1 25022681 Ki > 5290 nM T65019 CU6M9K 25060725 IC50 = 3100 nM T65019 CF7X2P 25060975 IC50 = 10500 nM T65019 CVR52U 25066764 IC50 = 1100 nM T65019 CD2KA4 25102047 IC50 = 94 nM T65019 CRW96X 25102048 IC50 = 95 nM T65019 CQ3O9P 25102050 IC50 = 41 nM T65019 CSHA26 25102051 IC50 = 81 nM T65019 C7ADO2 25102197 IC50 = 25 nM T65019 CA5DJ4 25138228 Ki = 4072000 nM T65019 C1TNQ3 25141117 Ki = 1900 nM T65019 CR35QP 25144971 IC50 > 10000 nM T65019 C0Y5BC 25145683 IC50 > 2500 nM T65019 CB7V8Y 25147773 IC50 = 0.32 nM T65019 C3KF1V 25178145 IC50 = 2.1 nM T65019 C8PMK7 25178356 IC50 > 100000 nM T65019 CG5Y2R 25178357 IC50 = 306 nM T65019 C4PZY6 25180866 IC50 = 353 nM T65019 CEP9Q2 25180867 IC50 = 3.9 nM T65019 C9HZG2 25181078 IC50 = 33900 nM T65019 CMYP34 25181079 IC50 = 8950 nM T65019 C7U1YC 25181080 IC50 = 89.8 nM T65019 C85HLG 25181081 IC50 = 260 nM T65019 CHR2P1 25183768 Ki > 25000 nM T65019 C6AR8O 42623563 IC50 > 100000 nM T65019 CX0VP7 42623564 IC50 = 52000 nM T65019 C0H3RD 42627769 IC50 = 6820 nM T65019 CPO1Z3 44123600 IC50 = 91 nM T65019 C25ELB 44143088 IC50 = 72443.6 nM T65019 CL0M7R 44143089 IC50 = 426579.52 nM T65019 C9QDC0 44143091 IC50 = 134896.29 nM T65019 CT80ED 44219901 IC50 = 3400 nM T65019 C94JVY 44219902 IC50 = 2800 nM T65019 C7J6GH 44219903 IC50 = 590 nM T65019 C9J7WL 44219904 IC50 = 11000 nM T65019 CRQ71E 44219905 IC50 = 6500 nM T65019 C4Z0ID 44219906 IC50 = 2400 nM T65019 CRNA25 44220092 IC50 > 1000 nM T65019 C9T5ZF 44220093 IC50 = 14000 nM T65019 CV38TE 44222825 IC50 = 5500 nM T65019 CJI73R 44222826 IC50 = 320 nM T65019 CGQ30N 44222827 IC50 = 1000 nM T65019 CCI64J 44224245 IC50 = 2250 nM T65019 CLRT69 44247751 IC50 = 33 nM T65019 CG7X5F 44272675 IC50 = 19.3 nM T65019 CEHR24 44272853 IC50 = 72 nM T65019 CJU31O 44321285 Ki = 73 nM T65019 C41VFA 44321286 Ki = 40 nM T65019 C5S2ZU 44321484 Ki = 545 nM T65019 CLQ23M 44321485 Ki = 192 nM T65019 CHF76Q 44321540 Ki = 45 nM T65019 CVOL49 44321593 Ki = 63 nM T65019 CB97GK 44321601 Ki = 90 nM T65019 CT0O7Y 44321602 Ki = 1282 nM T65019 CU62BP 44321746 Ki = 41 nM T65019 CQU2K9 44321782 Ki = 217 nM T65019 CV8T3N 44321783 Ki = 60 nM T65019 CIBO50 44321801 Ki = 22 nM T65019 C4E8GU 44321802 Ki = 125 nM T65019 CYDN18 44321803 Ki = 53 nM T65019 C7Z4DQ 44321887 Ki = 32 nM T65019 CFJ20T 44321932 Ki = 41 nM T65019 C9O0VB 44321965 Ki = 2960 nM T65019 C2E3RF 44321966 Ki = 271 nM T65019 CW9S1N 44321967 Ki = 1350 nM T65019 C1FI3O 44321975 Ki = 26 nM T65019 CLB8J6 44321976 Ki = 270 nM T65019 CR0KN1 44322209 Ki = 2030 nM T65019 C5LE1P 44322210 Ki = 92 nM T65019 CQ7AW8 44322211 Ki = 550 nM T65019 CJY2O7 44322214 Ki = 660 nM T65019 CR9GI0 44322215 Ki = 580 nM T65019 CMLA39 44329018 IC50 = 10 nM T65019 C1IE0S 44330147 IC50 > 100000 nM T65019 CE3MT4 44341611 Ki = 30100 nM T65019 CJTZ45 44341652 Ki = 30000 nM T65019 CTQ6P4 44344631 IC50 = 66900 nM T65019 CBH9I5 44344658 IC50 = 930 nM T65019 CGQ92A 44364037 IC50 = 62 nM T65019 C36YLM 44364111 IC50 = 835 nM T65019 CN4T7Q 44364119 IC50 = 521 nM T65019 CH4TE7 44364121 IC50 = 39 nM T65019 CPE91Y 44364122 IC50 = 52 nM T65019 CG2X0C 44364224 IC50 = 1102 nM T65019 C1F8XN 44364249 IC50 = 68 nM T65019 CWM47H 44364250 IC50 = 867 nM T65019 C0W5TL 44364251 IC50 = 20820 nM T65019 C3TPO7 44364266 IC50 = 4613 nM T65019 CJ2B8F 44364280 IC50 = 3108 nM T65019 CV0T6G 44383797 Ki = 9000 nM T65019 C9NIT7 44383842 Ki = 35000 nM T65019 C13LRY 44383990 Ki = 11000 nM T65019 CDQV80 44384020 Ki = 29000 nM T65019 CA2L3U 44384021 Ki = 15000 nM T65019 CT1MN8 44384090 Ki = 180000 nM T65019 CILQ34 44384272 Ki = 9500 nM T65019 CIJ61R 44384273 Ki = 14000 nM T65019 CL59ZH 44384393 Ki = 33000 nM T65019 C0RXF4 44384804 Ki = 1400 nM T65019 CE5RJ0 44385333 Ki = 20000 nM T65019 C5R4EW 44389591 IC50 > 300 nM T65019 C3EZ0W 44391336 IC50 = 50 nM T65019 C1E5JC 44391341 IC50 = 3 nM T65019 CT5Y1X 44391344 IC50 = 620 nM T65019 CP0QS3 44391345 IC50 = 27 nM T65019 CR0Y3D 44391350 IC50 = 16 nM T65019 CMTB94 44391351 IC50 = 70 nM T65019 CC7QW9 44391352 IC50 = 220 nM T65019 C0FC5U 44391354 IC50 = 11 nM T65019 CMS1Z6 44391356 IC50 = 18 nM T65019 CA3NH7 44391357 IC50 = 650 nM T65019 CTK65L 44391360 IC50 = 230 nM T65019 C0S4YB 44391365 IC50 = 120 nM T65019 CN4GJ0 44391366 IC50 = 9300 nM T65019 CKL09S 44391376 IC50 = 510 nM T65019 CVTB31 44391377 IC50 > 30000 nM T65019 C3BPI8 44391397 IC50 = 23 nM T65019 CW90KP 44391398 IC50 = 1400 nM T65019 C1N8KB 44391410 IC50 = 340 nM T65019 CB0HI5 44391419 IC50 = 23 nM T65019 C5XSH0 44391424 IC50 = 8700 nM T65019 CFH41S 44391425 IC50 = 18 nM T65019 C49DCW 44391434 IC50 = 60 nM T65019 CZ89IE 44391435 IC50 = 200 nM T65019 CP0AU9 44391440 IC50 = 260 nM T65019 C9BMR7 44391444 IC50 = 19 nM T65019 CR4U6B 44391445 IC50 = 75 nM T65019 CH59GY 44391449 IC50 = 150 nM T65019 CU7N6G 44391450 IC50 = 150 nM T65019 CD5TX3 44391460 IC50 = 6700 nM T65019 CCK39J 44391461 IC50 = 22 nM T65019 C3V1PB 44391476 IC50 = 36 nM T65019 C37DHM 44391486 IC50 = 220 nM T65019 CZB81D 44395506 IC50 = 83 nM T65019 CAU5R4 44397021 IC50 = 6600 nM T65019 CSO92L 44397377 IC50 = 1.5 nM T65019 CZ45GV 44397680 IC50 = 10900 nM T65019 C91POV 44402021 IC50 = 1490 nM T65019 CYCJ78 44402280 IC50 = 116 nM T65019 CY6WL5 44404502 IC50 = 12302.69 nM T65019 CWGQ46 44404503 IC50 = 15000 nM T65019 CLXM58 44404504 IC50 = 30000 nM T65019 C30DKN 44404553 IC50 = 4 nM T65019 CIC60V 44406452 IC50 = 3000 nM T65019 CVM7Y3 44413975 IC50 = 725 nM T65019 C4X0GA 44413977 IC50 = 488 nM T65019 CH01EO 44413978 IC50 = 891 nM T65019 CQ8HK9 44413979 IC50 = 4850 nM T65019 CBT0P2 44413982 IC50 = 583 nM T65019 CIJ39D 44413983 IC50 = 97 nM T65019 C9BA0V 44413987 IC50 = 1515 nM T65019 CE3WP0 44413991 IC50 = 5910 nM T65019 CDUI73 44413992 IC50 = 12 nM T65019 CH2X6W 44413997 IC50 = 1380 nM T65019 CHN85S 44414002 IC50 = 1900 nM T65019 C2OJ4B 44414029 IC50 = 2740 nM T65019 CT5PC9 44422672 IC50 = 11 nM T65019 CS9D5U 44422720 IC50 = 11 nM T65019 CNWM05 44422723 IC50 = 130 nM T65019 C58LAY 44422724 IC50 = 32 nM T65019 CDQU41 44422736 IC50 = 180 nM T65019 CVUB56 44422737 IC50 = 75 nM T65019 CB8G2W 44422743 IC50 = 26 nM T65019 CFX42T 44422744 IC50 = 6000 nM T65019 C9EL7F 44422749 IC50 = 40000 nM T65019 CO24JF 44423677 IC50 = 9500 nM T65019 C45WZX 44426073 IC50 = 1.6 ug.mL-1 T65019 CWU7G8 44434565 IC50 = 2660 nM T65019 CF9HU5 44434566 IC50 = 53100 nM T65019 CV3M6F 44434578 IC50 = 2490 nM T65019 CB9P0C 44442303 IC50 = 3440 nM T65019 C7HO0Y 44442304 IC50 = 7440 nM T65019 CAR3S2 44442305 IC50 = 3410 nM T65019 CZK0A9 44442306 IC50 = 4160 nM T65019 C71MCV 44442307 IC50 = 5640 nM T65019 CN70HO 44442308 IC50 = 1460 nM T65019 CVE5P0 44442309 IC50 = 5650 nM T65019 C3PT7N 44442310 IC50 = 1860 nM T65019 CGS18B 44442311 IC50 = 3020 nM T65019 CCFV76 44442313 IC50 = 5640 nM T65019 C4HYM6 44442314 IC50 = 1250 nM T65019 CZ2PE6 44442315 IC50 = 1650 nM T65019 C3I7RG 44442317 IC50 = 1020 nM T65019 CD9Y4Q 44445920 IC50 = 60.26 nM T65019 CL67QM 44445921 IC50 = 15.85 nM T65019 C6IS7V 44445922 IC50 = 18.2 nM T65019 CBL68C 44445923 IC50 = 120.23 nM T65019 C5Z4RH 44445924 IC50 = 512.86 nM T65019 CU9O6F 44445925 IC50 = 22.91 nM T65019 CWI9S1 44445926 IC50 = 50.12 nM T65019 CA6CX0 44445927 IC50 = 70.79 nM T65019 CQC1S9 44445928 IC50 = 19.05 nM T65019 C5GU9H 44445929 IC50 = 151.36 nM T65019 CX09NS 44445930 IC50 = 6760.83 nM T65019 C3XD8C 44445931 IC50 = 218.78 nM T65019 C6CPY9 44445932 IC50 = 199.53 nM T65019 CG0Z7I 44478924 IC50 = 4000 nM T65019 CFO27Y 44478926 IC50 = 200 nM T65019 CBZJ29 44478927 IC50 = 710 nM T65019 CRJ24K 44479197 IC50 = 360 nM T65019 CGOH82 44479198 IC50 = 8100 nM T65019 CLV56M 44479199 IC50 = 740 nM T65019 CY92OQ 44479458 IC50 = 120000 nM T65019 CH1QG9 44479459 IC50 = 1300 nM T65019 CB1NT7 44479460 IC50 = 940 nM T65019 C0JQ9L 44479699 IC50 = 860 nM T65019 C0DN1Q 44479700 IC50 = 77000 nM T65019 CTG24W 44479702 IC50 = 18000 nM T65019 CGZ49M 44479703 IC50 = 2100 nM T65019 CAK94X 44563337 IC50 = 1690 nM T65019 CSH4K3 44563364 IC50 > 10000 nM T65019 CAF95R 44563365 IC50 = 1000 nM T65019 CO4FQ1 44563366 IC50 > 10000 nM T65019 C6WA3X 44563401 IC50 > 10000 nM T65019 CX5L7N 44563402 IC50 = 2600 nM T65019 CJ8V4U 44563403 IC50 = 190 nM T65019 CN2BM4 44563404 IC50 = 3100 nM T65019 C3KCV6 44563405 IC50 = 3700 nM T65019 CI0R5M 44563465 IC50 = 1500 nM T65019 C5IQ9Z 44563466 IC50 = 1100 nM T65019 C6ZEW9 44563467 IC50 = 9700 nM T65019 CZ2EL1 44563468 IC50 = 5100 nM T65019 CDV6R7 44563469 IC50 = 730 nM T65019 CJ2BU5 44563487 IC50 = 10000 nM T65019 C1UXP6 44563490 IC50 = 105 nM T65019 CZ0W1A 44563491 IC50 = 3784 nM T65019 C4BD0N 44563493 IC50 = 1237 nM T65019 CNP6M7 44563494 IC50 = 2800 nM T65019 CWD32S 44580184 IC50 = 24000 nM T65019 CQ4ZR1 44580422 IC50 = 930 nM T65019 CK68GT 44580539 Ki = 67.6 nM T65019 CXIY57 44580801 Ki > 10000000 nM T65019 C0OA8Y 44580802 Ki > 10000000 nM T65019 CNC4D7 44581071 Ki > 10000000 nM T65019 CDF48U 44581111 Ki > 10000000 nM T65019 CTW7F2 44601281 IC50 = 41 nM T65019 C19LWR 44634267 IC50 = 23 nM T65019 CACH13 45269631 IC50 = 530 nM T65019 C36HRP 45377138 IC50 > 22000 nM T65019 C6B7ZY 45377564 IC50 > 500000 nM T65019 C5HAR6 45377565 IC50 > 22000 nM T65019 CKR0Q8 45377703 IC50 = 11000 nM T65019 C3SQL2 45378250 IC50 = 300 nM T65019 CQE49A 45378251 IC50 = 0.9 nM T65019 CO4AC6 45378252 IC50 = 210 nM T65019 C42FPG 45378253 IC50 = 4.3 nM T65019 CI82BN 45378254 IC50 = 29 nM T65019 C6MY2W 45380188 IC50 = 240 nM T65019 C9P0DG 45380189 IC50 = 16 nM T65019 CRY0E8 45380190 IC50 = 34 nM T65019 C0MPH3 45380191 IC50 = 1800 nM T65019 CMPE63 45482676 IC50 = 10000 nM T65019 CSX5I9 46175170 IC50 = 3.4 nM T65019 C56WVI 46184724 Ki > 30000 nM T65019 CDQ1K4 46224842 IC50 = 2.8 ug.mL-1 T65019 CH0Z1E 46844314 Ki = 1196 nM T65019 C20BTY 46856241 Ki = 1100 nM T65019 C5L8GF 46871738 IC50 > 10000 nM T65019 CR1KF7 46871739 IC50 = 5000 nM T65019 C8Q6YR 46871740 IC50 > 10000 nM T65019 C58YSM 46871741 IC50 > 10000 nM T65019 C4VEZ3 46882679 IC50 = 19 nM T65019 CR3QW7 46891107 IC50 > 10000 nM T65019 C5MK3A 46891108 IC50 > 10000 nM T65019 CQ5E1H 46891109 IC50 > 10000 nM T65019 C91LGI 46891170 IC50 = 2860 nM T65019 CZPM12 46891172 IC50 > 10000 nM T65019 C2V6MW 46891173 IC50 = 8220 nM T65019 C8S7QX 46891209 IC50 > 10000 nM T65019 C5Y0MN 46891255 IC50 > 10000 nM T65019 CJ16SE 46891256 IC50 > 10000 nM T65019 CNXU57 46891313 IC50 > 10000 nM T65019 CVK0E5 46891356 IC50 > 10000 nM T65019 C89RPO 46891357 IC50 > 10000 nM T65019 CVB6K4 46891358 IC50 > 10000 nM T65019 C0S9WB 46919610 Ki = 120 nM T65019 CE3H7I 46938726 IC50 = 1.33 nM T65019 C9T0HR 46938727 IC50 = 24.9 nM T65019 C0YR7M 46938728 IC50 = 7.1 nM T65019 C2TE8J 47162079 IC50 > 500000 nM T65019 CUD7O0 50941549 IC50 > 10000 nM T65019 CX8N4D 50990920 IC50 = 430 nM T65019 CXF4V3 50990921 IC50 > 8900 nM T65019 CAS94N 51346773 Ki = 480 nM T65019 CP65WT 51346774 Ki = 11000 nM T65019 C5OIA2 51346775 Ki = 32000 nM T65019 CU2SX3 51355576 Ki > 10000 nM T65019 CQM4E7 52936345 IC50 = 6.4 ug.mL-1 T65019 C1Y5UN 52951473 IC50 = 2200 nM T65019 CXYJ67 52951474 IC50 = 1400 nM T65019 C8J9EM 52951589 IC50 = 610 nM T65019 CEAS70 52951591 IC50 = 1100 nM T65019 C4DG1F 52951593 IC50 = 240 nM T65019 C6XJ3V 52951596 IC50 = 4900 nM T65019 C9U3AF 52951710 IC50 = 280 nM T65019 C4M1CA 52951712 IC50 = 4300 nM T65019 C76LDY 52951967 IC50 = 1.3 nM T65019 CYKS94 52951968 IC50 = 1.2 nM T65019 CE0FP3 52951969 IC50 = 100 nM T65019 CL69OM 52951970 IC50 = 100 nM T65019 CMPB74 52951971 IC50 = 17 nM T65019 CZ1TN8 52951972 IC50 = 8 nM T65019 CK08OB 52952074 IC50 = 25 nM T65019 C46AYR 52952075 IC50 = 450 nM T65019 CR32ZW 52952076 IC50 = 300 nM T65019 CJ9O3S 52952077 IC50 = 2100 nM T65019 C3N9TF 52952078 IC50 = 2500 nM T65019 C5S1IG 52952079 IC50 > 10000 nM T65019 CKV9R0 52952178 IC50 = 2900 nM T65019 CV0R6Y 52952179 IC50 = 6100 nM T65019 CE4Q7F 52952273 IC50 > 10000 nM T65019 CMA69V 52952274 IC50 = 6000 nM T65019 C7KB5W 52952275 IC50 = 5400 nM T65019 CRO0X4 52952276 IC50 = 1100 nM T65019 CSJ05E 52952277 IC50 = 1400 nM T65019 C29UJB 52952388 IC50 = 420 nM T65019 C3H5ID 52952389 IC50 = 270 nM T65019 CSX69R 52952390 IC50 = 2300 nM T65019 CB36KP 52952492 IC50 = 900 nM T65019 C67OEU 52952493 IC50 = 2100 nM T65019 CV1I0A 52952597 IC50 = 140 nM T65019 CGI87K 52952598 IC50 = 98 nM T65019 CXWI18 52952599 IC50 > 10000 nM T65019 C46VHP 52952600 IC50 = 2100 nM T65019 CH3G6R 52952601 IC50 > 10000 nM T65019 CC0Y3M 52952602 IC50 > 10000 nM T65019 CLA96C 53232689 Ki > 10000 nM T65019 C3BGW0 53233015 Ki > 40000 nM T65019 CMQZ70 53242178 IC50 > 23000 nM T65019 CRI92N 53311230 IC50 > 10000 nM T65019 C74CKF 53318123 Ki = 790 nM T65019 CB09MA 53318910 IC50 = 7.6 nM T65019 C47DIU 53318911 IC50 = 160 nM T65019 CC6DR2 53318912 IC50 = 4200 nM T65019 C7V1NC 53320225 IC50 = 4600 nM T65019 CVH2B7 53320226 IC50 > 18000 nM T65019 CO8QK2 53320227 IC50 > 3600 nM T65019 CNS3F2 53321542 IC50 = 3600 nM T65019 C1N2BX 53322876 IC50 = 390 nM T65019 CSYW40 53322877 IC50 > 8000 nM T65019 CGUC59 53322878 IC50 = 2600 nM T65019 C3QHA6 53322879 IC50 > 3700 nM T65019 CI3WL5 53323418 Ki = 20000 nM T65019 C1VNZ9 53324198 IC50 = 180 nM T65019 C0H7FQ 53324260 IC50 = 29000 nM T65019 CU7YG9 53325497 IC50 = 900 nM T65019 C4G1HK 53325498 IC50 = 18000 nM T65019 CO5L1I 53325499 IC50 = 17000 nM T65019 CZA03W 53326760 IC50 = 360 nM T65019 CM53CG 53326761 IC50 = 40000 nM T65019 CWR6T4 53326860 IC50 = 56 nM T65019 CPY02U 53327890 IC50 = 2100 nM T65019 CPGE80 53327891 IC50 = 1700 nM T65019 CLJ4G2 53328858 IC50 = 700 nM T65019 C4G3QL 53328859 IC50 = 1600 nM T65019 CX1TW0 53328860 IC50 = 112 nM T65019 C0ZX5G 53329215 IC50 = 6600 nM T65019 CSU52A 53329216 IC50 = 23000 nM T65019 CNB63X 53361475 IC50 = 9330 nM T65019 C6Y2EV 53374826 IC50 > 100000 nM T65019 CX3DU4 53378973 Ki = 12000 nM T65019 CTD1H9 53378974 Ki = 19000 nM T65019 C1IFJ8 53957122 IC50 > 500000 nM T65019 CSUW40 54352406 IC50 = 135 nM T65019 C3M8GZ 54580051 IC50 > 100000 nM T65019 CL0WM9 54580052 IC50 > 10000 nM T65019 CK26XF 54580053 IC50 > 10000 nM T65019 CS1LM9 54580054 IC50 = 226 nM T65019 C3LF0P 54580544 Ki > 10000 nM T65019 C6R3MZ 54580973 Ki > 50000 nM T65019 C8PE1G 54581030 IC50 = 2900 nM T65019 CVO09J 54581546 Ki > 10000 nM T65019 CWKA42 54582019 Ki > 50000 nM T65019 CVK72M 54582073 IC50 = 3100 nM T65019 CBK18O 54582074 IC50 > 10000 nM T65019 CP2F1B 54582075 IC50 > 10000 nM T65019 CZNU23 54582076 IC50 > 10000 nM T65019 C0U5HZ 54582077 IC50 > 7500 nM T65019 CSTG96 54582078 IC50 = 1400 nM T65019 C8SG9Y 54582079 IC50 > 10000 nM T65019 CZI6S3 54582080 IC50 > 7200 nM T65019 CD09BZ 54582543 Ki > 10000 nM T65019 CH6Q2Z 54583016 IC50 > 10000 nM T65019 C3V9LQ 54583017 IC50 = 1200 nM T65019 CT80KQ 54583018 IC50 > 770 nM T65019 CPT4L5 54583019 IC50 > 10000 nM T65019 CK52YD 54583511 Ki > 10000 nM T65019 CBEV27 54584024 IC50 > 10000 nM T65019 CM87DP 54584025 IC50 = 2900 nM T65019 C28GKQ 54585927 IC50 > 10000 nM T65019 CAZ76E 54586892 IC50 > 10000 nM T65019 CM0OQ3 54586893 IC50 > 10000 nM T65019 CK1NS7 54586894 IC50 > 10000 nM T65019 CMC4Y1 54586895 IC50 > 10000 nM T65019 C2MKX5 54586896 IC50 = 8000 nM T65019 CU91QP 54586897 IC50 > 10000 nM T65019 CI08RQ 54586898 IC50 > 10000 nM T65019 C6PRI4 54586899 IC50 > 10000 nM T65019 CG37UX 54587429 Ki > 10000 nM T65019 CL9SC3 54587769 Ki = 16400 nM T65019 C13FSJ 54669762 Ki = 210 nM T65019 CHS01Z 54669766 Ki = 28900 nM T65019 C7E9SG 54757202 Ki = 260 nM T65019 CKJ9S1 56835167 IC50 = 83 nM T65019 C21CLZ 56835168 IC50 = 3900 nM T65019 C0L2TS 56835169 IC50 = 2200 nM T65019 CKEV19 56850269 IC50 > 500000 nM T65019 C13DBR 56850270 IC50 > 500000 nM T65019 C05CTJ 56850271 IC50 = 51000 nM T65019 CX8QD5 56850272 IC50 = 225000 nM T65019 C1I9RE 56850407 IC50 > 500000 nM T65019 CVJ90W 56850408 IC50 = 15000 nM T65019 CPI5G0 56850409 IC50 = 41000 nM T65019 CHE2I1 57345500 Ki > 50000 nM T65019 C63TFM 57345501 Ki > 50000 nM T65019 C8KT2F 57345502 Ki > 50000 nM T65019 C0KPD8 57384084 IC50 = 160 nM T65019 CV67JB 57384091 IC50 = 3800 nM T65019 CN2H9K 57391204 IC50 > 10000 nM T65019 CR8MW2 57391205 IC50 > 10000 nM T65019 CNQ9B2 57392969 IC50 > 100000 nM T65019 CTYP14 57392972 IC50 > 10000 nM T65019 C5VB0U 57392973 IC50 > 10000 nM T65019 CMQL31 57392974 IC50 > 10000 nM T65019 C39OHF 57392975 IC50 > 10000 nM T65019 CDCW73 57394678 IC50 > 500000 nM T65019 CNOH63 57394711 IC50 > 10000 nM T65019 CD50CO 57399918 IC50 > 10000 nM T65019 CK68EY 57403424 IC50 > 10000 nM T65019 C0G2VY 57403564 IC50 = 5 nM T65019 CWH7V8 57561293 IC50 = 239 nM T65019 CY1N3J 57792153 IC50 = 1067 nM T65019 CCKD80 58307579 Ki = 62 nM T65019 C8ITK7 59794408 IC50 = 9501 nM T65019 CAT67H 59910477 IC50 = 1389 nM T65019 CH76IU 70684364 Ki = 190 nM T65019 CZ63AG 70684365 Ki = 280 nM T65019 C0GKT8 70685026 IC50 = 420 nM T65019 CTUN76 70688632 Ki = 580 nM T65019 C3LCG0 70688633 Ki = 140 nM T65019 C1A0VU 70692840 Ki = 5080 nM T65019 C6P3XM 70693710 Ki > 50000 nM T65019 CL7JF9 71304794 IC50 = 2200 nM T65019 CSY30R 71304795 IC50 = 250 nM T65019 CNPG78 71304796 IC50 = 1830 nM T65019 CMW3O0 71451330 Ki = 30000 nM T65019 CDZ3P2 71453147 Ki = 5100 nM T65019 C9QS6E 71456659 Ki = 105 nM T65019 CH5J4A 71602247 IC50 = 1600 nM T65019 CH53IU 71602248 IC50 = 4800 nM T65019 C97EWQ 71602249 IC50 = 4600 nM T65019 CNX9B1 71652215 IC50 = 82 nM T65019 C7RZN9 71652216 IC50 = 310 nM T65019 C0NTU7 71652382 IC50 = 24 nM T65019 CA5XS1 71652383 IC50 = 3700 nM T65019 C7DMX5 71680709 Ki = 11 nM T65019 CFPM82 71680710 Ki = 21 nM T65019 C9ZOM7 71680866 Ki = 6.6 nM T65019 CQ68LT 71680868 Ki = 85000 nM T65019 CV3X1T 71682766 Ki = 410 nM T65019 C5EAO8 71682767 Ki = 68 nM T65019 C80EYX 71682913 Ki = 3000 nM T65019 CIBD03 71682914 Ki = 1200 nM T65019 C41BYG 71682915 Ki = 18 nM T65019 C93XEI 71682916 Ki = 10 nM T65019 CQ29PJ 71682917 Ki > 200000 nM T65019 CFWN65 71683062 Ki > 25000 nM T65019 C3E2VT 71814508 IC50 = 671 nM T65019 CR2L4T 71814509 IC50 = 62 nM T65019 CF21LN 71814684 IC50 = 116 nM T65019 C4YM2D 71814685 IC50 = 915 nM T65019 CZW1P6 71814686 IC50 = 1080 nM T65019 C5SI6C 71814687 IC50 = 7731 nM T65019 CDXZ25 71814688 IC50 = 764 nM T65019 CIZ7K1 71814857 IC50 = 450 nM T65019 C4W9TJ 71814858 IC50 = 1282 nM T65019 CJH9K3 71814859 IC50 = 6897 nM T65019 CCMN52 71814860 IC50 = 4090 nM T65019 CZ9BC5 71814861 IC50 = 350 nM T65019 CU28BE 71815035 IC50 = 1858 nM T65019 C7HN2J 71815036 IC50 = 53584 nM T65019 CLWC38 72193198 IC50 = 100 nM T65019 CX4G0R 72204928 IC50 > 100000 nM T65019 CG9C6U 72204929 IC50 = 3900 nM T65019 C5A6XZ 72204930 IC50 = 26000 nM T65019 C0XZK4 72204931 IC50 > 100000 nM T65019 CM8Y7X 72204932 IC50 > 100000 nM T65019 C6RY4X 72204933 IC50 > 100000 nM T65019 C4N5AB 72204934 IC50 > 100000 nM T65019 C3H2FZ 72205111 IC50 > 100000 nM T65019 CQ0VX7 72205112 IC50 > 100000 nM T65019 CQ7TI1 72205113 IC50 = 43000 nM T65019 CPAW52 72205114 IC50 = 76000 nM T65019 C2LD3J 72205115 IC50 = 49500 nM T65019 CE4J8F 72711063 Ki = 1900 nM T65019 CW2RF1 72711064 Ki = 2100 nM T65019 CC5T1Q 72711065 Ki = 2500 nM T65019 C7YFC8 72711513 IC50 = 21400 nM T65019 CTM4P2 72713638 IC50 = 630 nM T65019 C0N2JX 72713639 IC50 = 590 nM T65019 CF4K8Y 72713862 IC50 = 7200 nM T65019 C3R6JO 72713863 IC50 = 72000 nM T65019 CW9D3V 72713864 IC50 = 1600 nM T65019 CQ6FH3 72713865 IC50 = 940 nM T65019 C4FYB0 72713866 IC50 = 2900 nM T65019 CH6SI1 72713867 IC50 = 1700 nM T65019 CS21QM 72713868 IC50 = 120000 nM T65019 CB56AP 72714081 IC50 = 890 nM T65019 C1CK0E 72714082 IC50 = 113000 nM T65019 CP5Q8W 72714083 IC50 = 123000 nM T65019 CRUH64 72714085 IC50 = 170000 nM T65019 COQZ24 72714091 Ki = 2400 nM T65019 CC0ZX4 72714092 Ki = 2700 nM T65019 CW8I1S 72714093 Ki = 2800 nM T65019 C3Q9LV 72714094 Ki = 3000 nM T65019 CZFY06 72714322 IC50 = 104000 nM T65019 CDY70J 72714323 IC50 = 68000 nM T65019 CD56BA 72714324 IC50 = 19500 nM T65019 CE51LQ 72714333 Ki = 17000 nM T65019 CK6D5F 72714334 Ki = 27000 nM T65019 C9FL7V 72714339 Ki = 2600 nM T65019 C38IDL 73345835 Ki = 7 nM T65019 CCV78D 73346037 IC50 > 99999 nM T65019 CK0TR7 73349097 IC50 = 98907 nM T65019 C57LGA 73349098 IC50 = 33882 nM T65019 C8ROG3 73350414 Ki = 6.2 nM T65019 CF7AB2 73350415 Ki = 70 nM T65019 C2PFM4 73351930 Ki = 310 nM T65019 CA2X8C 73352170 IC50 > 100000 nM T65019 CNW2C8 73353628 IC50 > 10000 nM T65019 CYV0L6 73353629 IC50 > 10000 nM T65019 CI09CY 73354906 Ki = 6 nM T65019 C1HLC9 73355128 IC50 > 10000 nM T65019 C06BPT 73355130 IC50 = 2817 nM T65019 C4SXT6 73356696 IC50 > 10000 nM T65019 CA5T7P 73603957 IC50 = 8000 nM T65019 C8VN1R 74221194 IC50 = 3900 nM T65019 C5LB0U 78426619 IC50 > 100000 nM T65019 CET6N8 78426757 IC50 > 100000 nM T65019 CUE7G4 86287514 IC50 > 50000 nM T65019 CGQ8F3 86287515 IC50 = 8700 nM T65019 CJ37XE 86287516 IC50 = 37000 nM T65019 COV8I9 86291010 IC50 = 1085 nM T65019 CO2FL5 90137145 IC50 = 3400 nM T65019 CRT54C 101910871 IC50 = 86000 nM T65019 C1J3CK 117094707 IC50 = 100000 nM T65019 C5ZS4E 118722686 IC50 = 3500 nM T65019 CIZB24 118722687 IC50 = 18000 nM T65019 C5C0ZX 118722688 IC50 = 8600 nM T65019 CLCW15 122181996 IC50 > 100000 nM T65019 CT7D4F 122181997 IC50 > 100000 nM T65019 CZO32N 122181998 IC50 > 100000 nM T65019 C40DWG 122181999 IC50 > 100000 nM T65019 CJFS09 122190237 IC50 = 5500 nM T65019 CT03QA 127026888 IC50 = 50000 nM T65019 C89QOM 127043503 IC50 = 6311 nM T65019 C9E5YJ 127043505 IC50 = 1614 nM T65019 CW1Q3D 127043506 IC50 = 5424 nM T65019 C1C7WB 127044036 IC50 = 6875 nM T65019 CPF6U7 127044139 IC50 = 7783 nM T65019 CT9B0Q 127044462 IC50 = 4639 nM T65019 CL3X1A 127044649 IC50 = 8805 nM T65019 C8RZ7T 127044651 IC50 = 1000 nM T65019 C3I4PT 127044652 IC50 = 807 nM T65019 CDX86T 127044818 IC50 = 2407 nM T65019 C56OJV 127044819 IC50 = 427 nM T65019 CYA92R 130282633 IC50 = 6500 nM T65019 CO3QE2 130282636 IC50 = 4400 nM T65019 C4MB7N 132285189 Ki = 120 nM T65019 CTN42D 132941363 IC50 = 78000 nM T65019 CT3G2U 134133460 IC50 = 23 nM T65019 C8VLY0 134144890 IC50 = 850 nM T65019 C93ZLI 134145328 IC50 = 900 nM T65019 CHV2U1 135438561 IC50 > 10000 nM T65019 C4FVJ1 135487604 IC50 > 100000 nM T65019 C1MOD4 135567320 IC50 > 10000 nM T65019 CA5JR6 136054481 IC50 > 10000 nM T65019 CV47JN 136054485 IC50 = 8900 nM T65019 CZ48WO 136054487 IC50 > 10000 nM T65019 C8FGT0 136054495 IC50 = 3700 nM T65019 CG70BZ 136054516 IC50 = 5.4 nM T65019 CSM57W 136054520 IC50 = 550 nM T65019 CJG54U 136219136 IC50 > 30000 nM T65019 C3CAV5 136219141 IC50 = 24000 nM T65019 CPB07Z 136241630 IC50 = 4300 nM T65019 CIEW62 136380958 IC50 = 140 nM T65019 C9HS7J 137287436 IC50 = 3.8 nM T65019 C4UMY5 137636781 IC50 > 5000 nM T65019 CR8H9Z 137644167 IC50 > 5000 nM T65019 CB8M6U 137646865 IC50 > 5000 nM T65019 CK4LE6 137647628 IC50 > 10000 nM T65019 CS80YI 137652598 IC50 = 1600 nM T65019 CZB75K 137657128 IC50 > 10000 nM T65019 CC3I9B 137660260 IC50 > 10000 nM T65019 C4H0EM 137661370 IC50 > 5000 nM T65019 CZ8H6N 137661550 IC50 = 7600 nM T65019 C37HMX 137701229 Ki = 53 nM T65019 C1Q2BP 145949247 IC50 > 5000 nM T65019 C6TD4M 145949288 IC50 > 5000 nM T65019 CN9RD6 145949408 IC50 > 5000 nM T65019 C5FWA2 145949488 IC50 > 5000 nM T65019 CZS1N7 145949693 IC50 > 5000 nM T65019 C6IPV3 145949783 IC50 = 435800 nM T65019 CYG32L 145950058 IC50 > 5000 nM T65019 C72LGN 145950074 IC50 > 500000 nM T65019 CU53BP 145950331 IC50 > 5000 nM T65019 CY8C4A 145950332 IC50 > 5000 nM T65019 CAJ25P 145951291 IC50 > 5000 nM T65019 C3EF7N 145952515 IC50 > 5000 nM T65019 CW1GS2 145952760 IC50 > 5000 nM T65019 CFN1R7 145952843 IC50 > 5000 nM T65019 CM6T2O 145953417 IC50 > 5000 nM T65019 C6FYK8 145953609 IC50 > 5000 nM T65019 CV80WQ 145954107 IC50 > 5000 nM T65019 C16VNH 145954604 IC50 > 5000 nM T65019 CQF50V 145954863 IC50 > 5000 nM T65019 C2HAG8 145955226 IC50 = 309300 nM T65019 C8QW9G 145955776 IC50 > 5000 nM T65019 CH0ZO5 145955778 IC50 > 5000 nM T65019 CFDZ62 145955866 IC50 > 5000 nM T65019 CVZ5U7 145955868 IC50 > 5000 nM T65019 C8TPR1 145956198 IC50 > 5000 nM T65019 COR96H 145956298 IC50 = 301100 nM T65019 CR8U7Y 145956318 IC50 > 5000 nM T65019 C7R3FE 145956426 IC50 = 76300 nM T65019 C4S8LU 145956764 IC50 > 5000 nM T65019 CUS0Y9 145957234 IC50 > 5000 nM T65019 CUO69Q 145957392 IC50 > 5000 nM T65019 CX94UK 145957493 IC50 > 5000 nM T65019 C6MHN7 145957508 IC50 > 5000 nM T65019 CQ15DP 145957734 IC50 = 111350 nM T65019 C5K7PV 145958060 IC50 > 5000 nM T65019 CBE02W 145958354 IC50 > 5000 nM T65019 CQL4O0 145959327 IC50 > 5000 nM T65019 CG03OE 145959777 IC50 = 109000 nM T65019 CIQ9J2 145960035 IC50 = 87100 nM T65019 CUAT97 145960347 IC50 > 5000 nM T65019 CZ76WA 145962290 IC50 > 5000 nM T65019 C27MTZ 145962695 IC50 > 5000 nM T65019 CRY63E 145963538 IC50 > 5000 nM T65019 CVCL61 145963739 IC50 > 5000 nM T65019 CFE1A5 145971595 Ki = 119 nM T65019 CWY5X0 145971805 IC50 = 4000 nM T65019 C1FPG2 145972660 IC50 > 5000 nM T65019 CJF73O 145973630 IC50 > 5000 nM T65019 CX7M9L 145976456 IC50 > 5000 nM T65019 C1KPL5 145976497 IC50 = 40000 nM T65019 CPD1B0 145977213 IC50 > 5000 nM T65019 C9Z5DX 145978402 IC50 > 5000 nM T65019 CZ25LW 155512044 IC50 = 57000 nM T65019 C98HMU 155515777 IC50 = 80 nM T65019 CRY3D4 155541376 IC50 = 14 nM T65019 CH40UO 155562232 IC50 = 7 nM T65019 CP9YX2 155567218 IC50 = 26000 nM T65019 C8D5VK 155567855 IC50 = 34000 nM T65019 CLT4Y6 10138589 Ki = 290 nM T65019 D01UNE 44580457 Ki = 160 nM T65019 D03AMR 9849669 Ki = 1200 nM T65019 D04GOO 10111838 IC50 > 100000 nM T65019 D04PAW 16216218 IC50 = 70000 nM T65019 D04VPH 45376872 IC50 = 8300 nM T65019 D05THD 44478925 IC50 = 8300 nM T65019 D06EHW 11625778 IC50 = 772 nM T65019 D06HSC 136117931 IC50 = 80000 nM T65019 D07DRT 46175162 Ki = 4 nM T65019 D07GEL 10344307 Ki = 94 nM T65019 D07MJD 44479701 IC50 = 5400 nM T65019 D09USO 5277466 IC50 = 40000 nM T65019 D09ZOA 25049753 IC50 = 70 nM T65019 D0A0FY 44479457 IC50 = 25000 nM T65019 D0A4TC 446504 IC50 = 7.5 nM T65019 D0B3UN 44580458 Ki = 140 nM T65019 D0G3YZ 11391583 IC50 = 36600 nM T65019 D0H6CK 10160968 Ki > 5290 nM T65019 D0L4EO 11609208 IC50 = 30600 nM T65019 D0L6ND 10089677 IC50 = 0.2 ug.mL-1 T65019 D0NP8A 10370504 IC50 = 1900 nM T65019 D0NV9C 22004198 IC50 = 360 nM T65019 D0P2TS 9818682 IC50 > 10000 nM T65019 D0Q4TA 10044321 IC50 = 2300 nM T65019 D0S9OL 10155934 IC50 = 1300 nM T65019 D0W2UK 6914621 Ki = 15872 nM T65019 D0XK7G 10445302 IC50 = 210 nM T65019 D0Y5IQ 44255320 IC50 = 5000 nM T39919 D00BCP 2727 IC50 = 133000 nM T39919 D00BLL 9849808 IC50 = 133000 nM T39919 D00DKK 5282379 IC50 = 133000 nM T39919 D00FGO 460612 IC50 = 133000 nM T39919 D00IBN 54676228 IC50 = 133000 nM T39919 D00JAU 3749 IC50 = 83200 nM T39919 D00KVO 2082 IC50 = 133000 nM T39919 D00MIN 657298 IC50 = 133000 nM T39919 D00NKB 5546 IC50 = 133000 nM T39919 D00USF 5533 IC50 = 133000 nM T39919 D00WAM 3647 IC50 = 133000 nM T39919 D00WUF 5486971 IC50 = 133000 nM T39919 D00XUN 23894 IC50 = 133000 nM T39919 D00YZA 5453 IC50 = 133000 nM T39919 D01AJY 2284 IC50 = 133000 nM T39919 D01AZG 5073 IC50 = 133000 nM T39919 D01DBQ 452548 IC50 = 34900 nM T39919 D01GBY 124087 IC50 = 133000 nM T39919 D01KKQ 135400182 IC50 = 133000 nM T39919 D01MDT 5487 IC50 = 133000 nM T39919 D01MUR 68844 IC50 = 133000 nM T39919 D01OXI 2578 IC50 = 133000 nM T39919 D01STB 5362129 IC50 = 133000 nM T39919 D01UTL 2995 IC50 = 133000 nM T39919 D01UXC 2249 IC50 = 133000 nM T39919 D01XNB 4594 IC50 = 133000 nM T39919 D01XYJ 35370 IC50 = 133000 nM T39919 D01ZII 2726 IC50 = 133000 nM T39919 D01ZSO 4235 IC50 = 133000 nM T39919 D02DGU 444795 IC50 = 133000 nM T39919 D02DPA 2756 IC50 = 133000 nM T39919 D02FEM 5284447 IC50 = 133000 nM T39919 D02HED 4748 IC50 = 133000 nM T39919 D02LCR 5467 IC50 = 133000 nM T39919 D02NTO 5510 IC50 = 133000 nM T39919 D02STN 132971 IC50 = 133000 nM T39919 D02TLO 3690 IC50 = 133000 nM T39919 D02YIZ 12560 IC50 = 133000 nM T39919 D02ZTJ 5339 IC50 = 1500 nM T39919 D03CQE 5379 IC50 = 133000 nM T39919 D03DDR 3034034 IC50 = 133000 nM T39919 D03ELL 2159 IC50 = 133000 nM T39919 D03HJK 447043 IC50 = 133000 nM T39919 D03JSJ 446596 IC50 = 133000 nM T39919 D03KOZ 1549120 IC50 = 6500 nM T39919 D03KQF 4011 IC50 = 133000 nM T39919 D03KZM 216237 IC50 = 133000 nM T39919 D03NHW 4583 IC50 = 133000 nM T39919 D03QWT 73303 IC50 = 133000 nM T39919 D03RTS 2662 IC50 = 133000 nM T39919 D03TVW 54120 IC50 = 133000 nM T39919 D03TYI 9433 IC50 = 131000 nM T39919 D03VPC 2754 IC50 = 16600 nM T39919 D03XOC 656583 IC50 = 133000 nM T39919 D03YLZ 27200 IC50 = 133000 nM T39919 D04AAW 60613 IC50 = 133000 nM T39919 D04ASH 657180 IC50 = 133000 nM T39919 D04EGX 54746 IC50 = 133000 nM T39919 D04FBR 5281078 IC50 = 83000 nM T39919 D04ITO 6436173 IC50 = 30200 nM T39919 D04JCN 47811 IC50 = 133000 nM T39919 D04JEE 4946 IC50 = 133000 nM T39919 D04JPJ 3950 IC50 = 133000 nM T39919 D04KYY 135401907 IC50 = 133000 nM T39919 D04MSM 2554 IC50 = 133000 nM T39919 D04NXQ 51081 IC50 = 133000 nM T39919 D04OSE 4485 IC50 = 16600 nM T39919 D04RGA 5282415 IC50 = 7100 nM T39919 D04VMT 5253 IC50 = 133000 nM T39919 D04WFD 4543 IC50 = 133000 nM T39919 D04XGT 31593 IC50 = 133000 nM T39919 D04YMH 151166 IC50 = 133000 nM T39919 D04ZTY 444020 IC50 = 133000 nM T39919 D05AFX 4450 IC50 = 133000 nM T39919 D05ARP 135398740 IC50 = 133000 nM T39919 D05DVP 5717 IC50 = 12100 nM T39919 D05EAM 4735 IC50 = 133000 nM T39919 D05FTJ 4044 IC50 = 133000 nM T39919 D05GJW 20279 IC50 = 133000 nM T39919 D05HPI 16134395 IC50 = 133000 nM T39919 D05HSC 6000 IC50 = 9600 nM T39919 D05LEO 3385 IC50 = 133000 nM T39919 D05LKP 5215 IC50 = 133000 nM T39919 D05LYX 3488 IC50 = 10500 nM T39919 D05MFA 135398741 IC50 = 133000 nM T39919 D05MQK 110635 IC50 = 133000 nM T39919 D05OFX 219078 IC50 = 133000 nM T39919 D05QDC 5284513 IC50 = 49000 nM T39919 D05UVD 33624 IC50 = 133000 nM T39919 D05VIL 5284594 IC50 = 133000 nM T39919 D05VIX 3463 IC50 = 133000 nM T39919 D05VLS 5090 IC50 = 133000 nM T39919 D05ZGQ 5281070 IC50 = 133000 nM T39919 D05ZIK 4205 IC50 = 133000 nM T39919 D06ABF 3957 IC50 = 133000 nM T39919 D06BEP 2712 IC50 = 133000 nM T39919 D06CTE 57469 IC50 = 133000 nM T39919 D06FDR 135398739 IC50 = 133000 nM T39919 D06GAM 3357 IC50 = 133000 nM T39919 D06GDY 43815 IC50 = 133000 nM T39919 D06HBQ 91610 IC50 = 6300 nM T39919 D06JPB 5280793 IC50 = 133000 nM T39919 D06NXY 5991 IC50 = 133000 nM T39919 D06OIV 5505 IC50 = 133000 nM T39919 D06OMK 445643 IC50 = 133000 nM T39919 D06OVY 5362065 IC50 = 133000 nM T39919 D06PSS 5311309 IC50 = 133000 nM T39919 D06TNL 3278 IC50 = 133000 nM T39919 D06UDG 60846 IC50 = 133000 nM T39919 D06WTZ 53232 IC50 = 133000 nM T39919 D06XAE 1712095 IC50 = 24500 nM T39919 D06XMU 6013 IC50 = 133000 nM T39919 D06YYD 9578005 IC50 = 133000 nM T39919 D06ZII 969472 IC50 = 133000 nM T39919 D06ZUK 3696 IC50 = 133000 nM T39919 D07ABV 468595 IC50 = 133000 nM T39919 D07BCT 36294 IC50 = 133000 nM T39919 D07CWD 3657 IC50 = 133000 nM T39919 D07DJQ 10219 IC50 = 133000 nM T39919 D07GRH 2749 IC50 = 133000 nM T39919 D07HGR 5362119 IC50 = 133000 nM T39919 D07HVY 64139 IC50 = 133000 nM T39919 D07IEF 2391 IC50 = 133000 nM T39919 D07IPB 454216 IC50 = 36800 nM T39919 D07JGT 4421 IC50 = 57500 nM T39919 D07JVL 3016 IC50 = 133000 nM T39919 D07KSG 2733526 IC50 = 133000 nM T39919 D07QCE 2265 IC50 = 133000 nM T39919 D07SUG 2478 IC50 = 133000 nM T39919 D07TQV 60825 IC50 = 133000 nM T39919 D07UBG 130881 IC50 = 28500 nM T39919 D07UYO 441401 IC50 = 133000 nM T39919 D07VDZ 5284627 IC50 = 133000 nM T39919 D07VLY 31703 IC50 = 19000 nM T39919 D07WEP 3019 IC50 = 133000 nM T39919 D07XGR 3339 IC50 = 133000 nM T39919 D07XSN 6253 IC50 = 133000 nM T39919 D08EBN 41684 IC50 = 133000 nM T39919 D08HVR 6047 IC50 = 133000 nM T39919 D08IWD 57363 IC50 = 51000 nM T39919 D08JIV 2162 IC50 = 133000 nM T39919 D08PIQ 6741 IC50 = 40970 nM T39919 D08QIP 4887 IC50 = 2700 nM T39919 D08QMX 5757 IC50 = 133000 nM T39919 D08ROP 3899 IC50 = 133000 nM T39919 D08USJ 4456 IC50 = 133000 nM T39919 D08VRO 3822 IC50 = 133000 nM T39919 D08VXL 5353788 IC50 = 133000 nM T39919 D08VYV 4168 IC50 = 133000 nM T39919 D08ZEB 2733 IC50 = 133000 nM T39919 D09CZA 5282226 IC50 = 74000 nM T39919 D09DHY 6167 IC50 = 133000 nM T39919 D09DWL 5719 IC50 = 133000 nM T39919 D09EGZ 2719 IC50 = 103900 nM T39919 D09HNR 3002190 IC50 = 7100 nM T39919 D09HVL 16129704 IC50 = 133000 nM T39919 D09IOI 2170 IC50 = 133000 nM T39919 D09IPV 28417 IC50 = 133000 nM T39919 D09JUG 60490 IC50 = 133000 nM T39919 D09LNI 3365 IC50 = 133000 nM T39919 D09LWS 150311 IC50 = 133000 nM T39919 D09MGR 123619 IC50 = 53000 nM T39919 D09NIA 2732 IC50 = 133000 nM T39919 D09QEI 4740 IC50 = 133000 nM T39919 D09TBD 5344 IC50 = 133000 nM T39919 D09WEJ 2446 IC50 = 133000 nM T39919 D09XQF 3767 IC50 = 133000 nM T39919 D09XZB 123631 IC50 = 4600 nM T39919 D0A0OO 65016 IC50 = 133000 nM T39919 D0A2ZX 4173 IC50 = 133000 nM T39919 D0A5SE 134018 IC50 = 1900 nM T39919 D0A9YA 6918296 IC50 = 133000 nM T39919 D0AA2D 2378 IC50 = 133000 nM T39919 D0AD5C 41774 IC50 = 133000 nM T39919 D0AN7B 896 IC50 = 133000 nM T39919 D0AO5H 5578 IC50 = 133000 nM T39919 D0AP9T 53025 IC50 = 133000 nM T39919 D0AV3G 3151 IC50 = 133000 nM T39919 D0AZ3C 5291 IC50 = 133000 nM T39919 D0B1IP 5282375 IC50 = 133000 nM T39919 D0B2GI 3476 IC50 = 64000 nM T39919 D0B2UZ 4917 IC50 = 133000 nM T39919 D0B3HD 2519 IC50 = 133000 nM T39919 D0B5MP 135398513 IC50 = 133000 nM T39919 D0B6TW 135403647 IC50 = 133000 nM T39919 D0B7EB 36462 IC50 = 133000 nM T39919 D0B7NG 2725 IC50 = 133000 nM T39919 D0B8UJ 3011155 IC50 = 133000 nM T39919 D0BA9U 13109 IC50 = 133000 nM T39919 D0BM5G 5381 IC50 = 133000 nM T39919 D0C3YQ 23662354 IC50 = 133000 nM T39919 D0C4RB 36314 IC50 = 133000 nM T39919 D0C6NM 5311221 IC50 = 133000 nM T39919 D0C8EU 5394 IC50 = 133000 nM T39919 D0CL9S 159269 IC50 = 133000 nM T39919 D0CT9C 2907 IC50 = 133000 nM T39919 D0CW1P 9782 IC50 = 133000 nM T39919 D0D0BE 28061 IC50 = 133000 nM T39919 D0D0ZD 441314 IC50 = 133000 nM T39919 D0D1AL 3559 IC50 = 133000 nM T39919 D0D1SG 5755 IC50 = 133000 nM T39919 D0D2VS 60198 IC50 = 133000 nM T39919 D0D4JO 6917864 IC50 = 133000 nM T39919 D0D5GD 3373 IC50 = 133000 nM T39919 D0D5GG 4723 IC50 = 133000 nM T39919 D0D7KC 5488548 IC50 = 133000 nM T39919 D0D7LA 4091 IC50 = 133000 nM T39919 D0D8XY 5311010 IC50 = 133000 nM T39919 D0DJ1B 156391 IC50 = 133000 nM T39919 D0E0SW 53708 IC50 = 133000 nM T39919 D0E1SW 1986 IC50 = 133000 nM T39919 D0E1XL 5284583 IC50 = 133000 nM T39919 D0E6OC 5282230 IC50 = 1000 nM T39919 D0E6XR 3062316 IC50 = 27300 nM T39919 D0E6YQ 1935 IC50 = 23700 nM T39919 D0E7PQ 5311 IC50 = 133000 nM T39919 D0EG1I 9926791 IC50 = 133000 nM T39919 D0EJ6O 2763 IC50 = 133000 nM T39919 D0ES1Q 6918289 IC50 = 44000 nM T39919 D0F2PO 4828 IC50 = 133000 nM T39919 D0F6EO 33613 IC50 = 133000 nM T39919 D0F7CS 6758 IC50 = 133000 nM T39919 D0F8RA 2153 IC50 = 133000 nM T39919 D0F9GE 3108 IC50 = 8300 nM T39919 D0FM2P 82153 IC50 = 133000 nM T39919 D0G3DL 135398735 IC50 = 41900 nM T39919 D0G4OD 54686904 IC50 = 133000 nM T39919 D0G5AG 104762 IC50 = 133000 nM T39919 D0G5UB 2161 IC50 = 2200 nM T39919 D0G7FJ 54677470 IC50 = 133000 nM T39919 D0G8NN 119570 IC50 = 133000 nM T39919 D0G9IU 135403821 IC50 = 35900 nM T39919 D0G9YH 2179 IC50 = 7430 nM T39919 D0GU4K 135413536 IC50 = 133000 nM T39919 D0GY5Z 2244 IC50 = 133000 nM T39919 D0H0KB 5070 IC50 = 133000 nM T39919 D0H0ND 54454 IC50 = 133000 nM T39919 D0H3HM 60795 IC50 = 133000 nM T39919 D0H3WI 37542 IC50 = 133000 nM T39919 D0H6QU 6005 IC50 = 133000 nM T39919 D0H8FH 3702 IC50 = 133000 nM T39919 D0I0EG 44093 IC50 = 133000 nM T39919 D0I2MK 4171 IC50 = 133000 nM T39919 D0I4DQ 5280723 IC50 = 2300 nM T39919 D0I6IB 54677971 IC50 = 133000 nM T39919 D0I7SZ 54892 IC50 = 133000 nM T39919 D0IT2G 5743 IC50 = 133000 nM T39919 D0IT2X 2581 IC50 = 3000 nM T39919 D0J1MI 4030 IC50 = 15500 nM T39919 D0J1VY 5281081 IC50 = 6800 nM T39919 D0J2KV 4932 IC50 = 133000 nM T39919 D0J2MJ 26758 IC50 = 133000 nM T39919 D0J4JM 5770 IC50 = 133000 nM T39919 D0J5DC 2796 IC50 = 133000 nM T39919 D0JC9N 60164 IC50 = 133000 nM T39919 D0JO7Y 104741 IC50 = 133000 nM T39919 D0JV4Q 3002820 IC50 = 133000 nM T39919 D0JY3V 107751 IC50 = 133000 nM T39919 D0K0OZ 5702160 IC50 = 133000 nM T39919 D0K0VO 5639 IC50 = 133000 nM T39919 D0K3MC 3947 IC50 = 133000 nM T39919 D0K3QS 6442177 IC50 = 95000 nM T39919 D0K5CB 2083 IC50 = 133000 nM T39919 D0K6GZ 60464 IC50 = 133000 nM T39919 D0K7HU 6918155 IC50 = 133000 nM T39919 D0K7WK 4595 IC50 = 133000 nM T39919 D0K8KX 5280343 IC50 = 20800 nM T39919 D0KG3R 9875401 IC50 = 133000 nM T39919 D0KR2J 135398508 IC50 = 133000 nM T39919 D0L3DK 6918537 IC50 = 133000 nM T39919 D0L5RW 65015 IC50 = 133000 nM T39919 D0L5WM 2157 IC50 = 133000 nM T39919 D0L6DA 119607 IC50 = 133000 nM T39919 D0L7FM 4911 IC50 = 133000 nM T39919 D0L9ZR 4891 IC50 = 133000 nM T39919 D0M2MR 3475 IC50 = 133000 nM T39919 D0M3QP 441207 IC50 = 133000 nM T39919 D0M4YC 3114 IC50 = 133000 nM T39919 D0M5JI 9560989 IC50 = 133000 nM T39919 D0M5OC 5484727 IC50 = 133000 nM T39919 D0M6DO 2145 IC50 = 133000 nM T39919 D0M8RC 5403 IC50 = 133000 nM T39919 D0M8VE 71360 IC50 = 133000 nM T39919 D0M9BW 68911 IC50 = 133000 nM T39919 D0M9DC 4614 IC50 = 12000 nM T39919 D0MA9N 2955 IC50 = 133000 nM T39919 D0ML1F 60871 IC50 = 133000 nM T39919 D0N0RU 82146 IC50 = 133000 nM T39919 D0N0TZ 60606 IC50 = 133000 nM T39919 D0N1FS 26248 IC50 = 6400 nM T39919 D0N3VR 71616 IC50 = 133000 nM T39919 D0N4OW 644077 IC50 = 133000 nM T39919 D0N5HJ 5462501 IC50 = 133000 nM T39919 D0N5YA 65981 IC50 = 53900 nM T39919 D0N6RF 65999 IC50 = 36000 nM T39919 D0NG7O 60857 IC50 = 133000 nM T39919 D0NJ3V 4680 IC50 = 23130 nM T39919 D0NR6S 3002977 IC50 = 133000 nM T39919 D0NS6H 3152 IC50 = 72900 nM T39919 D0NW3X 71329 IC50 = 133000 nM T39919 D0O1WX 2764 IC50 = 133000 nM T39919 D0O2EM 4463 IC50 = 133000 nM T39919 D0O2SR 47528 IC50 = 133000 nM T39919 D0O3OS 104850 Ki = 4000 nM T39919 D0O4SE 5479 IC50 = 133000 nM T39919 D0O5FY 441130 IC50 = 133000 nM T39919 D0O5WP 148124 IC50 = 133000 nM T39919 D0OB1J 39186 IC50 = 133000 nM T39919 D0OT0O 44561 IC50 = 133000 nM T39919 D0P1UX 5656 IC50 = 133000 nM T39919 D0P7JZ 34359 IC50 = 133000 nM T39919 D0P9RF 5401 IC50 = 36800 nM T39919 D0PQ3G 3440 IC50 = 133000 nM T39919 D0PW7C 51039 IC50 = 133000 nM T39919 D0Q2PE 4539 IC50 = 133000 nM T39919 D0Q2XF 5311027 IC50 = 133000 nM T39919 D0Q3YO 1547484 IC50 = 133000 nM T39919 D0Q4SD 443872 IC50 = 133000 nM T39919 D0Q4XQ 3291 IC50 = 133000 nM T39919 D0Q4YK 4843 IC50 = 133000 nM T39919 D0Q5NX 216326 IC50 = 133000 nM T39919 D0Q5UQ 214348 IC50 = 36500 nM T39919 D0Q6NZ 5281034 IC50 = 133000 nM T39919 D0Q8ZX 2337 IC50 = 133000 nM T39919 D0QL3P 34312 IC50 = 133000 nM T39919 D0R0BX 6604200 IC50 = 20900 nM T39919 D0R0FE 2520 IC50 = 133000 nM T39919 D0R1RS 3715 IC50 = 5800 nM T39919 D0R1WR 4919 IC50 = 133000 nM T39919 D0R2KJ 18381 IC50 = 133000 nM T39919 D0R3FP 6398764 IC50 = 133000 nM T39919 D0R3QY 5665 IC50 = 133000 nM T39919 D0R5RR 119182 IC50 = 133000 nM T39919 D0R7HO 2471 IC50 = 133000 nM T39919 D0R8ER 3229 IC50 = 133000 nM T39919 D0R9OH 5329 IC50 = 133000 nM T39919 D0R9VR 9651 IC50 = 133000 nM T39919 D0S1NZ 5310993 IC50 = 133000 nM T39919 D0S3WH 68827 IC50 = 133000 nM T39919 D0S4BR 1349907 IC50 = 133000 nM T39919 D0S5CU 4499 IC50 = 16500 nM T39919 D0S5UH 2794 IC50 = 44500 nM T39919 D0S5WG 3366 IC50 = 133000 nM T39919 D0S9MC 2789 IC50 = 133000 nM T39919 D0S9SD 60877 IC50 = 133000 nM T39919 D0SH3I 387447 IC50 = 133000 nM T39919 D0SV8E 126941 IC50 = 133000 nM T39919 D0T0KA 4474 IC50 = 88000 nM T39919 D0T1LK 4908 IC50 = 133000 nM T39919 D0T2PL 5280453 IC50 = 133000 nM T39919 D0T2XU 4927 IC50 = 133000 nM T39919 D0T5WK 4506 IC50 = 133000 nM T39919 D0T7US 5281037 IC50 = 133000 nM T39919 D0T8GD 89594 IC50 = 133000 nM T39919 D0T8VY 71771 IC50 = 133000 nM T39919 D0T9DT 2140 IC50 = 133000 nM T39919 D0T9TJ 3034010 IC50 = 133000 nM T39919 D0TR5X 3386 IC50 = 133000 nM T39919 D0U0KW 208902 IC50 = 133000 nM T39919 D0U1OM 60726 IC50 = 133000 nM T39919 D0U2JP 4369359 IC50 = 133000 nM T39919 D0U4CE 104865 IC50 = 22000 nM T39919 D0U4UQ 3639 IC50 = 133000 nM T39919 D0U5GB 92727 IC50 = 47000 nM T39919 D0U5QK 1983 IC50 = 133000 nM T39919 D0U5RT 4909 IC50 = 133000 nM T39919 D0U5SI 4913 IC50 = 133000 nM T39919 D0U8UV 10660 IC50 = 133000 nM T39919 D0UF6M 9568512 IC50 = 133000 nM T39919 D0UL2L 54690031 IC50 = 133000 nM T39919 D0UM7O 3821 IC50 = 133000 nM T39919 D0V4QS 135398745 IC50 = 133000 nM T39919 D0V7CF 5362440 IC50 = 133000 nM T39919 D0V8QT 2708 IC50 = 133000 nM T39919 D0V9BD 2375 IC50 = 133000 nM T39919 D0VM2L 68740 IC50 = 133000 nM T39919 D0VT8P 3324 IC50 = 133000 nM T39919 D0W0BF 2187 IC50 = 133000 nM T39919 D0W9LX 2585 IC50 = 133000 nM T39919 D0WI3T 441243 IC50 = 59000 nM T39919 D0WN0U 3333 IC50 = 133000 nM T39919 D0WS1X 6915944 IC50 = 11600 nM T39919 D0WV3U 4893 IC50 = 12500 nM T39919 D0X0RI 4178 IC50 = 133000 nM T39919 D0X3FX 5284596 IC50 = 133000 nM T39919 D0X4RN 3676 IC50 = 133000 nM T39919 D0X5SD 3117 IC50 = 133000 nM T39919 D0X5XU 451668 IC50 = 133000 nM T39919 D0X6GN 444025 IC50 = 133000 nM T39919 D0X6IU 5959 IC50 = 133000 nM T39919 D0X7DE 4449 IC50 = 71000 nM T39919 D0X7KZ 6918182 IC50 = 133000 nM T39919 D0X7XG 3000226 IC50 = 133000 nM T39919 D0X9RG 5361092 IC50 = 133000 nM T39919 D0X9ZC 47965 IC50 = 133000 nM T39919 D0XF8W 1046 IC50 = 133000 nM T39919 D0Y0SW 3397 IC50 = 133000 nM T39919 D0Y2CJ 4201 IC50 = 133000 nM T39919 D0Y3MO 37768 IC50 = 133000 nM T39919 D0Y5DO 2771 IC50 = 133000 nM T39919 D0Y5UG 2160 IC50 = 133000 nM T39919 D0Y7EM 3332 IC50 = 8200 nM T39919 D0Y7IU 5281004 IC50 = 37000 nM T39919 D0Y7PG 4659569 IC50 = 16700 nM T39919 D0Y7ZU 135398738 IC50 = 133000 nM T39919 D0Y9LL 42884 IC50 = 133000 nM T39919 D0YV1Q 6032 IC50 = 133000 nM T39919 D0Z1RV 135398737 IC50 = 133000 nM T39919 D0Z1ZM 84029 IC50 = 133000 nM T39919 D0Z3DY 2333 IC50 = 17000 nM T39919 D0Z4EI 55245 IC50 = 133000 nM T39919 D0Z4SB 3478 IC50 = 133000 nM T39919 D0Z4UN 6509979 IC50 = 133000 nM T39919 D0Z4ZT 68873 IC50 = 37900 nM T39919 D0Z5BC 5634 IC50 = 63900 nM T39919 D0Z5IU 1548887 IC50 = 133000 nM T39919 D0Z6UC 5358 IC50 = 133000 nM T39919 D0Z7KE 3784 IC50 = 133000 nM T39919 D0Z8EX 18283 IC50 = 133000 nM T39919 D0Z9QR 24066 IC50 = 133000 nM T39919 D0ZB7K 5735 IC50 = 133000 nM T39919 D0ZS8P 2801 IC50 = 133000 nM T39919 D0ZU9R 392622 IC50 = 34000 nM T39919 D00TIG 6917964 IC50 = 133000 nM T39919 D08YWK 6436 IC50 = 133000 nM T39919 D09YDM 24360 IC50 = 7400 nM T39919 D0E3TC 44259 IC50 = 37900 nM T39919 D0G7UX 5284373 IC50 = 133000 nM T39919 D0Q9CY 9915743 IC50 = 23000 nM T39919 D0SD9V 53276 IC50 = 133000 nM T39919 D0TO2R 30751 IC50 = 133000 nM T39919 D0VG0D 11977753 IC50 = 133000 nM T39919 D0Y1FO 472335 IC50 = 5100 nM T39919 D01PIL 54477 IC50 = 133000 nM T39919 D01VAB 2119 IC50 = 133000 nM T39919 D02LHR 33625 IC50 = 133000 nM T39919 D03JPH 54677972 IC50 = 133000 nM T39919 D04BQR 4342 IC50 = 133000 nM T39919 D05RUM 15387 IC50 = 133000 nM T39919 D06ABW 2788 IC50 = 133000 nM T39919 D07XPE 8249 IC50 = 133000 nM T39919 D08SOF 5405 IC50 = 133000 nM T39919 D0C0JT 4495 IC50 = 133000 nM T39919 D0G9ZW 54676478 IC50 = 133000 nM T39919 D0J9GD 64715 IC50 = 133000 nM T39919 D0O2IE 4754 IC50 = 133000 nM T39919 D0OS6O 60149 IC50 = 133000 nM T39919 D0P1JI 312145 IC50 = 63200 nM T39919 D0S6QR 214350 IC50 = 133000 nM T39919 D0T1RG 216235 IC50 = 28400 nM T39919 D0Y2HR 2247 IC50 = 133000 nM T39919 D0Y4FL 6915744 IC50 = 133000 nM T39919 D0Y8UB 82148 IC50 = 133000 nM T39919 C85KQB 2202 IC50 = 133000 nM T39919 CI74WY 2450 IC50 = 133000 nM T39919 CPJ0C2 2747 IC50 = 133000 nM T39919 C36WOC 2800 IC50 = 133000 nM T39919 C7CT6M 2804 IC50 = 133000 nM T39919 CJ0B9F 3158 IC50 = 133000 nM T39919 C0H8GR 3191 IC50 = 133000 nM T39919 CEXU05 3383 IC50 = 133000 nM T39919 COSX53 3519 IC50 = 133000 nM T39919 CO2Y3R 3698 IC50 = 133000 nM T39919 C4ZJT8 3730 IC50 = 133000 nM T39919 CY4WG9 3793 IC50 = 133000 nM T39919 C9LCD8 3823 IC50 = 69000 nM T39919 C2KJI7 3883 IC50 = 133000 nM T39919 C12UDR 4411 IC50 = 133000 nM T39919 C8VXJ6 4888 IC50 = 9800 nM T39919 C93BJO 5039 IC50 = 133000 nM T39919 C5N0SU 5334 IC50 = 133000 nM T39919 C48GPY 5475 IC50 = 133000 nM T39919 C1EYR7 5497 IC50 = 133000 nM T39919 C2U1WA 6216 IC50 = 133000 nM T39919 C59UQE 6279 IC50 = 22500 nM T39919 CC09DB 9703 IC50 = 133000 nM T39919 CO1I7C 11080 IC50 = 133000 nM T39919 CMU2P6 11683 IC50 = 133000 nM T39919 C2J7BV 12947 IC50 = 133000 nM T39919 CVJ2X3 14051 IC50 = 133000 nM T39919 C6RG5E 21233 IC50 = 133000 nM T39919 CJ3OL7 25590 IC50 = 133000 nM T39919 CK21BO 27350 IC50 = 133000 nM T39919 C4VU9Z 31098 IC50 = 133000 nM T39919 CUJ6W7 35455 IC50 = 133000 nM T39919 CZA2C6 39764 IC50 = 133000 nM T39919 CFX82C 47320 IC50 = 133000 nM T39919 C6E5CD 48229 IC50 = 133000 nM T39919 CE8LA7 49659 IC50 = 133000 nM T39919 CU86VK 54459 IC50 = 133000 nM T39919 C7ZUJ4 54840 IC50 = 133000 nM T39919 CC10UB 56801 IC50 = 133000 nM T39919 CQSF39 57004 IC50 = 133000 nM T39919 CH8GS0 60749 IC50 = 133000 nM T39919 CYQ4S7 60822 IC50 = 88500 nM T39919 CHZJ65 60834 IC50 = 133000 nM T39919 C2GKD5 62884 IC50 = 133000 nM T39919 CY8ES4 62935 IC50 = 133000 nM T39919 CA9S6G 62978 IC50 = 8000 nM T39919 C7SO5H 63021 IC50 = 133000 nM T39919 CP8F7B 64143 IC50 = 97000 nM T39919 CD9TC8 64737 IC50 = 133000 nM T39919 C7WUM6 65335 IC50 = 133000 nM T39919 COZ10X 65348 IC50 = 133000 nM T39919 CS7L6J 65957 IC50 = 133000 nM T39919 C7AV1G 68553 IC50 = 133000 nM T39919 C73LEV 71399 IC50 = 133000 nM T39919 C6A4VW 71651 IC50 = 133000 nM T39919 C2F1OT 77997 IC50 = 133000 nM T39919 C1W8YJ 78000 IC50 = 133000 nM T39919 C6NLX4 84003 IC50 = 2700 nM T39919 CVP7G8 101526 IC50 = 133000 nM T39919 C90TYQ 130313 IC50 = 133000 nM T39919 CAR7Y4 146571 IC50 = 133000 nM T39919 C3WVZ6 154068 IC50 = 133000 nM T39919 CI7BE6 219025 IC50 = 133000 nM T39919 CA6ID2 241903 IC50 = 35100 nM T39919 CV80FO 249332 IC50 = 133000 nM T39919 C0VN3D 288216 IC50 = 133000 nM T39919 CLD6J9 441074 IC50 = 45800 nM T39919 CY7HM4 441313 IC50 = 133000 nM T39919 CDU0B1 441351 IC50 = 133000 nM T39919 CVX0K8 443866 IC50 = 133000 nM T39919 C40YBS 444036 IC50 = 133000 nM T39919 C35HJB 656684 IC50 = 133000 nM T39919 CGIY90 688272 IC50 = 133000 nM T39919 CBM17N 3000706 IC50 = 133000 nM T39919 C4BR7C 3005572 IC50 = 133000 nM T39919 CWQI02 3033817 IC50 = 133000 nM T39919 CH86TV 3033968 IC50 = 133000 nM T39919 C2XP0H 3052775 IC50 = 133000 nM T39919 CONV41 4022878 IC50 = 133000 nM T39919 C4SL8Q 5281025 IC50 = 133000 nM T39919 C9QDT1 5281067 IC50 = 133000 nM T39919 CNI9X4 5281888 IC50 = 6000 nM T39919 C4X7RJ 5282408 IC50 = 133000 nM T39919 C10CPM 5282455 IC50 = 26800 nM T39919 CBLX43 5282481 IC50 = 133000 nM T39919 CB4P2S 5289394 IC50 = 133000 nM T39919 CG53MU 5353627 IC50 = 133000 nM T39919 CUA96S 5388961 IC50 = 133000 nM T39919 C5DV8U 5702270 IC50 = 68200 nM T39919 C4GST2 6321416 IC50 = 28000 nM T39919 CC9WJ2 6433334 IC50 = 133000 nM T39919 CQR03B 6526396 IC50 = 133000 nM T39919 C0P8LZ 6602611 IC50 = 133000 nM T39919 CPK20Z 6917733 IC50 = 133000 nM T39919 C9FQ0W 6918092 IC50 = 133000 nM T39919 C9P2HT 9556529 IC50 = 133000 nM T39919 CEO67P 9588170 IC50 = 73200 nM T39919 C5W7MS 9833407 IC50 = 133000 nM T39919 CJL94H 9839243 IC50 = 133000 nM T39919 C7QK8R 9847786 IC50 = 133000 nM T39919 CIWP56 9886273 IC50 = 46000 nM T39919 C5NH4J 9912089 IC50 = 133000 nM T39919 C45JHO 9933004 IC50 = 133000 nM T39919 CIV15Q 10113978 IC50 = 8100 nM T39919 CZ1XW6 10483360 IC50 = 13500 nM T39919 C8BL9W 10695961 IC50 = 24000 nM T39919 CV2E4Z 11476710 IC50 = 34100 nM T39919 CVG4M1 11679357 IC50 = 133000 nM T39919 CZ6PB5 12001375 IC50 = 133000 nM T39919 CCLY36 12004215 IC50 = 133000 nM T39919 C9N5YG 14720269 IC50 = 133000 nM T39919 CGL5Q2 16051965 IC50 = 35600 nM T39919 CA3JL7 16052011 IC50 = 133000 nM T39919 C7WI4H 16204922 IC50 = 133000 nM T39919 CLHO84 16759173 IC50 = 133000 nM T39919 C71VGO 16760285 IC50 = 133000 nM T39919 CUZE40 18004026 IC50 = 133000 nM T39919 C28AYI 18530292 IC50 = 8080 nM T39919 C0REQ9 20055509 IC50 = 133000 nM T39919 CQ31BP 23623618 IC50 = 133000 nM T39919 CFE9R6 23666879 IC50 = 133000 nM T39919 CH59NC 23667631 IC50 = 133000 nM T39919 CWB0H2 23674512 IC50 = 133000 nM T39919 CFLN18 23675322 IC50 = 54200 nM T39919 CD01LT 23685176 IC50 = 133000 nM T39919 C9YI0H 23716436 IC50 = 1900 nM T39919 C3N4GQ 25078429 IC50 = 133000 nM T39919 CW7ZK4 44181971 IC50 = 133000 nM T39919 C4OT7Z 44403122 Ki = 7000 nM T39919 CUA6N3 46783232 IC50 = 133000 nM T39919 C9SCG4 49800073 IC50 = 133000 nM T39919 CRV3P5 54685920 IC50 = 133000 nM T39919 CGK7Y9 54685925 IC50 = 133000 nM T39919 CQ6C4E 56972143 IC50 = 2700 nM T39919 CM5T1V 57393422 IC50 = 133000 nM T39919 CTO71V 72734347 IC50 = 133000 nM T39919 CRZ62F 73355036 IC50 = 133000 nM T39919 C41TDB 135413523 IC50 = 26800 nM T39919 CDN1S3 135413539 IC50 = 133000 nM T39919 CG8C4T 135415564 IC50 = 15900 nM T39919 C27TMO 137648451 IC50 = 7500 nM T39919 CHPC06 137654606 IC50 = 133000 nM T39919 C67IKZ 145948937 IC50 = 133000 nM T39919 C9RLJ3 3661 IC50 = 133000 nM T39919 D01BJB 15032 IC50 = 133000 nM T39919 D01OIK 155774 IC50 = 133000 nM T39919 D03IRR 2206 IC50 = 133000 nM T39919 D04LBT 14957 IC50 = 133000 nM T39919 D07GXY 4850 IC50 = 133000 nM T39919 D08CNS 3748 IC50 = 133000 nM T39919 D09XCX 5694 IC50 = 44900 nM T39919 D0F4QX 5601 IC50 = 133000 nM T39919 D0F5LH 4634 IC50 = 133000 nM T39919 D0J6JT 1355 IC50 = 133000 nM T39919 D0L9PX 5943 IC50 = 133000 nM T39919 D0T5RO 16129706 IC50 = 133000 nM T39231 D01SHZ 9931954 IC50 = 144 nM T39231 D04AIT 5280445 IC50 = 2398.83 nM T39231 D0J9HW 23725625 IC50 = 1230 nM T39231 D00BMF 24958200 IC50 = 2344.23 nM T39231 D0F5TD 135565981 IC50 = 50 nM T39231 C3S7DE 1686 IC50 = 313 nM T39231 CH62DB 1853 IC50 = 112.2 nM T39231 CM82AL 51459 IC50 > 10000 nM T39231 CXG7Y0 76959 IC50 > 100000 nM T39231 CO7Z4L 77793 IC50 = 71 nM T39231 CS74HZ 145726 IC50 = 230 nM T39231 CNVB16 146013 IC50 > 10000 nM T39231 CW9I1J 146492 IC50 > 10000 nM T39231 C4FEY6 147157 IC50 > 10000 nM T39231 CW78JD 151515 IC50 = 233 nM T39231 C0F1IA 229015 IC50 = 310 nM T39231 C7ER4A 229016 IC50 = 794.33 nM T39231 CJ2UB5 236501 IC50 > 100000 nM T39231 C3PS2M 249526 IC50 > 10000 nM T39231 CY65EM 261391 IC50 = 275.42 nM T39231 C2O7DN 265714 IC50 = 360 nM T39231 C8AX6O 466268 IC50 = 5000 nM T39231 CYC75Z 622510 IC50 = 66 nM T39231 CH8FK7 1091861 IC50 = 15848.93 nM T39231 CA6OJ3 1241435 IC50 = 66.07 nM T39231 C40IBK 1506320 IC50 = 398.11 nM T39231 C6EZY0 1511413 IC50 = 251.19 nM T39231 C89WXS 2802462 IC50 = 6 nM T39231 C1HJR0 2817216 IC50 > 10000 nM T39231 CZ07RY 2817491 IC50 = 7 nM T39231 CTO30U 2825267 IC50 > 10000 nM T39231 C48HET 2825269 IC50 = 272 nM T39231 C1NOK3 2946601 IC50 = 1800 nM T39231 CZ8H1N 2959509 IC50 = 1000 nM T39231 CLJ6X7 3163516 IC50 = 630.96 nM T39231 CR26SK 4163640 IC50 = 1100 nM T39231 CT9V6M 4826644 IC50 = 620 nM T39231 C8ZW6Y 5272796 IC50 = 851.14 nM T39231 C4C8BV 5320693 IC50 = 560 nM T39231 CB86MY 5391140 IC50 = 280 nM T39231 C7CIL3 6490174 IC50 > 100000 nM T39231 C4P2UQ 8607850 IC50 > 100000 nM T39231 CAV3P4 9899130 IC50 = 199.53 nM T39231 CI0QP9 11960529 IC50 = 10740 nM T39231 C4Y5DW 12402280 IC50 = 90 nM T39231 CZ0KO4 14668434 IC50 = 31 nM T39231 CO9U6A 14735886 IC50 = 162 nM T39231 C5ZW8I 15989803 IC50 = 1258.93 nM T39231 CCBV16 16013151 IC50 = 1761 nM T39231 CG5A7W 16013152 IC50 = 2550 nM T39231 CPG4V1 16013160 IC50 = 559 nM T39231 CJ2XS5 16031314 IC50 = 395 nM T39231 C9LT3B 16031344 IC50 = 299 nM T39231 C80PHC 16193211 IC50 = 125.89 nM T39231 C4T7EK 16516470 IC50 = 1010 nM T39231 CZ6M5I 22431503 IC50 = 125.89 nM T39231 CO81DU 22432629 IC50 = 31.62 nM T39231 CP9H4Y 22432631 IC50 = 50.12 nM T39231 C0DW5F 22582935 IC50 = 28 nM T39231 CA3TO2 22582936 IC50 = 32 nM T39231 C1Y2MX 24772013 IC50 = 2000 nM T39231 CL8Q0K 24772834 IC50 = 3500 nM T39231 C0IOR9 25015515 IC50 = 3090.3 nM T39231 CMXA39 28825277 IC50 > 100000 nM T39231 CSO1Z6 28825295 IC50 > 100000 nM T39231 C8BKV6 44381234 IC50 = 407.38 nM T39231 CNI3Y5 44483163 IC50 = 131 nM T39231 CEI70H 45116983 IC50 = 144.54 nM T39231 C92MLH 46261432 IC50 = 19.95 nM T39231 C46BCE 46742374 IC50 = 114 nM T39231 C2XI7M 46742375 IC50 = 146 nM T39231 CWF40I 56587957 IC50 = 343 nM T39231 C6O1UZ 58829329 IC50 = 150 nM T39231 CN8AS7 67072266 IC50 > 100000 nM T39231 CD3HT9 67960134 IC50 = 46 nM T39231 C2JKD9 69004309 IC50 > 100000 nM T39231 C7QLY3 71464718 IC50 = 200 nM T39231 C24XZF 71576800 IC50 = 860 nM T39231 CED5V6 71622125 IC50 = 691.83 nM T39231 CI0GU8 71660496 IC50 = 2 nM T39231 CAO96N 71680699 IC50 > 20000 nM T39231 CI98LH 71680701 IC50 = 1300 nM T39231 C40RSX 71680702 IC50 > 20000 nM T39231 CHOZ71 71680703 IC50 = 4300 nM T39231 CL20JN 71680704 IC50 = 1500 nM T39231 CBH64M 71680705 IC50 = 400 nM T39231 C91BGF 71680860 IC50 = 1220 nM T39231 COP6V9 71680863 IC50 = 18 nM T39231 CBS20R 71681023 IC50 = 16 nM T39231 C1KT7H 71681028 IC50 = 10 nM T39231 CH1FS9 71681175 IC50 = 4 nM T39231 CZ1H8S 71681176 IC50 = 4 nM T39231 CCAK12 71681177 IC50 = 3 nM T39231 CHO50K 71681178 IC50 = 11 nM T39231 CJO9X1 71681179 IC50 = 1 nM T39231 CJ34PZ 71681180 IC50 = 4 nM T39231 C2RGP3 71681329 IC50 = 3 nM T39231 CI5E8F 71681330 IC50 = 1 nM T39231 C32RCL 71681331 IC50 = 143 nM T39231 CVJ86T 71681485 IC50 = 4 nM T39231 CY12QO 71681487 IC50 = 4 nM T39231 CH4V6D 71681649 IC50 = 5 nM T39231 CC0UX4 71683057 IC50 > 20000 nM T39231 CGU79X 71683058 IC50 > 20000 nM T39231 CX0M7D 71683059 IC50 > 20000 nM T39231 CFM05A 71683060 IC50 = 1600 nM T39231 C1MP6Q 71683061 IC50 = 540 nM T39231 C7KNH4 71736275 IC50 = 364 nM T39231 CL2H7E 71736276 IC50 = 16 nM T39231 C82YZD 71736278 IC50 = 12 nM T39231 CZS9B1 71736279 IC50 = 12 nM T39231 C2B5MQ 71736447 IC50 = 17 nM T39231 CF5M7C 71736755 IC50 = 13 nM T39231 CMJY69 71737385 IC50 = 17 nM T39231 CO96XF 71819164 IC50 = 262 nM T39231 CMC2J4 72193935 IC50 = 49 nM T39231 CL73DQ 72549316 IC50 = 7.943 nM T39231 CX9BU6 72549541 IC50 = 6.31 nM T39231 C06VKU 72549782 IC50 = 316.23 nM T39231 C46DHU 72724967 IC50 = 9 nM T39231 C8SL4X 72724968 IC50 = 148 nM T39231 CL3J2U 73056614 IC50 = 24 nM T39231 C8DX4G 73293052 IC50 = 14 nM T39231 CK67DZ 73293053 IC50 = 12 nM T39231 CE4PM3 73293055 IC50 = 7 nM T39231 CVTK56 73295340 IC50 = 31 nM T39231 CTWE30 73347820 IC50 = 64000 nM T39231 CNIH86 73351951 IC50 = 1250 nM T39231 CK9X5R 73356483 IC50 = 24 nM T39231 CU3D9N 73388373 IC50 = 2.512 nM T39231 C1OUQ4 73441895 IC50 = 19.95 nM T39231 CZY9U8 73441896 IC50 = 15.85 nM T39231 CR5E3W 73441897 IC50 = 10 nM T39231 CKF92G 73442057 IC50 = 25.12 nM T39231 CC51JH 73442058 IC50 = 3.981 nM T39231 C10MTI 73442172 IC50 = 15.85 nM T39231 CZKO04 73442173 IC50 = 25.12 nM T39231 CKGD48 73442233 IC50 = 7.943 nM T39231 CRO8S1 73442292 IC50 = 15.85 nM T39231 C6QO3Z 73442409 IC50 = 199.53 nM T39231 C1UQI4 73442411 IC50 = 125.89 nM T39231 CSP08U 73442462 IC50 = 398.11 nM T39231 CE8H9P 73442464 IC50 = 50.12 nM T39231 CS9H2V 73442467 IC50 = 19.95 nM T39231 C67FWO 73442584 IC50 = 100 nM T39231 CTUM58 73442643 IC50 = 7.943 nM T39231 CH18VD 73442700 IC50 = 10 nM T39231 C7YZ6G 73442705 IC50 = 63.1 nM T39231 CH3AT1 76280996 IC50 = 6.1 nM T39231 CZ7OL0 76284556 IC50 = 59 nM T39231 C8IT9R 76684090 IC50 = 133.3 nM T39231 CRE2U3 77050682 IC50 > 10000 nM T39231 C9VP6T 86276157 IC50 = 12 nM T39231 C3XO5D 89649815 IC50 = 562.34 nM T39231 C83KNV 89661926 IC50 = 1122.02 nM T39231 CL5RS1 90082725 IC50 = 25.12 nM T39231 C2EFL0 91810427 IC50 = 136 nM T39231 CF8W2B 91928421 IC50 = 19000 nM T39231 C2XR5Q 92045137 IC50 = 9 nM T39231 CV0NZ7 105539834 IC50 = 550 nM T39231 CYQ1E2 117999828 IC50 = 35 nM T39231 COD65L 117999906 IC50 = 18 nM T39231 CLZ1U3 118498201 IC50 = 0.18 nM T39231 CT78JM 118498266 IC50 = 0.2 nM T39231 C1VB9L 118507411 IC50 = 0.24 nM T39231 CI70KV 118717515 IC50 = 181 nM T39231 CRK45H 122177906 IC50 = 245.47 nM T39231 C8GS6E 122177907 IC50 = 331.13 nM T39231 C9SXK6 122177908 IC50 = 700 nM T39231 CH3RJ2 122177909 IC50 = 346.74 nM T39231 CL4A3P 122177910 IC50 = 570 nM T39231 C0ZKD7 122177911 IC50 = 4600 nM T39231 CP1QU7 122177912 IC50 = 2454.71 nM T39231 CVCS41 122177963 IC50 = 370 nM T39231 CDX95C 122177964 IC50 = 290 nM T39231 CYWJ91 122177965 IC50 = 290 nM T39231 CWO65I 122205439 IC50 = 483 nM T39231 C5QD0E 122205440 IC50 = 104 nM T39231 C02SDC 122423373 IC50 = 3200 nM T39231 CF2NO9 127037410 IC50 = 10964.78 nM T39231 CV06MU 131801402 IC50 = 28.84 nM T39231 CD1R6Q 135400456 IC50 = 1406 nM T39231 C9PI7O 135402338 IC50 = 1100 nM T39231 C0HQF2 135404247 IC50 = 140 nM T39231 C95RAN 135405744 IC50 = 528 nM T39231 C6FY0X 135416131 IC50 = 786 nM T39231 C6DBN7 135417258 IC50 = 346 nM T39231 CCY9H6 135417291 IC50 = 53 nM T39231 C1KBX6 135417551 IC50 = 135 nM T39231 C1PE8H 135417609 IC50 = 35 nM T39231 C47LAF 135418940 IC50 = 10 nM T39231 CIS9K5 135421564 IC50 = 224 nM T39231 CM5Q1Z 135430309 IC50 = 67 nM T39231 C4MW7F 135443732 IC50 = 299 nM T39231 CH14EB 135443955 IC50 = 5 nM T39231 C8XI3K 135448518 IC50 = 430 nM T39231 CZ9GA7 135449434 IC50 > 100000 nM T39231 CA0R7X 135452109 IC50 = 346 nM T39231 C9H1VA 135456692 IC50 = 1284 nM T39231 C8J2PC 135456762 IC50 = 48 nM T39231 CHY9C3 135479130 IC50 = 781 nM T39231 CJO81C 135513650 IC50 = 156 nM T39231 C7G6BQ 135513721 IC50 = 73 nM T39231 CU3FW2 135566794 IC50 = 8 nM T39231 C8QDG3 135566882 IC50 = 0.1 nM T39231 CVD04P 135566883 IC50 = 63 nM T39231 CNVM21 135566884 IC50 = 0.1 nM T39231 C4BFY3 135566969 IC50 = 35 nM T39231 C59OUK 135566970 IC50 = 50 nM T39231 C7K5WL 135566971 IC50 = 2423 nM T39231 CN74FK 135566972 IC50 = 153 nM T39231 CRY12I 135566973 IC50 = 22 nM T39231 CU2I7X 135567125 IC50 = 9.12 nM T39231 C37PTU 135567126 IC50 = 5.1 nM T39231 CT1DZ8 135644892 IC50 = 39.4 nM T39231 C38XBR 135652704 IC50 = 20.5 nM T39231 C1G4CE 135741330 IC50 = 93 nM T39231 CAT50N 135741861 IC50 = 485 nM T39231 C4ZGO7 135741892 IC50 = 110 nM T39231 CIL7K3 135742498 IC50 = 322 nM T39231 CS83CJ 135905416 IC50 = 100 nM T39231 C12CPN 136165102 IC50 = 1090 nM T39231 C54NVS 136175126 IC50 = 0.81 nM T39231 CVH7R6 136175127 IC50 = 8.5 nM T39231 CS5PH8 136175128 IC50 = 0.4 nM T39231 CY94ZB 136215772 IC50 = 36 nM T39231 C7JEG1 136215773 IC50 = 44 nM T39231 CF7O2U 136215774 IC50 = 73 nM T39231 CFP0V5 136215897 IC50 = 32 nM T39231 C18GVR 136224209 IC50 = 0.2 nM T39231 C80BWX 136224210 IC50 = 0.2 nM T39231 CBQ6R1 136224211 IC50 = 0.2 nM T39231 C0HS5P 136224212 IC50 = 400 nM T39231 CB19RP 136227775 IC50 = 155 nM T39231 CM4PB2 136236970 IC50 = 12.5 nM T39231 C50JYC 136236972 IC50 = 14 nM T39231 C1WG3C 136236974 IC50 = 17 nM T39231 CF1H5N 136236975 IC50 = 23 nM T39231 CU17IT 136236976 IC50 = 11 nM T39231 C71FDZ 136236977 IC50 = 10 nM T39231 CCL4D6 136236978 IC50 = 24 nM T39231 C9WHB4 136236979 IC50 = 3.3 nM T39231 C68GON 136236980 IC50 = 12 nM T39231 C18MSY 136236981 IC50 = 10 nM T39231 CF01JX 136236982 IC50 = 7 nM T39231 CYF2I1 136236983 IC50 = 1000 nM T39231 C3ZW8J 136236994 IC50 = 1.6 nM T39231 CN0J1C 136236995 IC50 = 35 nM T39231 CHJ8I2 136236997 IC50 = 1.2 nM T39231 C0LB6W 136236998 IC50 = 0.8 nM T39231 CVB4D7 136237000 IC50 = 26 nM T39231 CSB3Y1 136237004 IC50 = 1.5 nM T39231 C4H8ZN 136237010 IC50 = 15 nM T39231 CCL4V0 136240108 IC50 = 0.2 nM T39231 CHM35F 136240109 IC50 = 0.1 nM T39231 C8E0AF 136241425 IC50 = 800 nM T39231 CW17FT 136241426 IC50 = 27 nM T39231 C5NI6F 136241427 IC50 > 46000 nM T39231 CRWN30 136241639 IC50 = 0.2 nM T39231 C2KO4C 136241640 IC50 = 31 nM T39231 C52DUR 136241641 IC50 = 16 nM T39231 CFA4R8 136241642 IC50 = 1 nM T39231 CR07BF 136244504 IC50 = 5000 nM T39231 CHSN59 136245073 IC50 = 907 nM T39231 C7VX4R 136245086 IC50 = 21 nM T39231 CM5JC2 136245087 IC50 > 46000 nM T39231 CCIV06 136245088 IC50 > 46000 nM T39231 C3NX2H 136249376 IC50 = 0.2 nM T39231 C3RIV5 136249377 IC50 = 0.3 nM T39231 CE2I0N 136249378 IC50 = 0.2 nM T39231 CNOA16 136249379 IC50 = 1750 nM T39231 C5REV1 136249380 IC50 = 860 nM T39231 C3IQ7P 136249381 IC50 > 46000 nM T39231 C2P5LK 136253145 IC50 = 50 nM T39231 CHD0B7 136264278 IC50 = 2 nM T39231 C5DAO8 136264279 IC50 = 210 nM T39231 CCE28N 136264280 IC50 = 400 nM T39231 C2YO7J 136264281 IC50 = 640 nM T39231 C0D8MZ 136264443 IC50 = 46 nM T39231 C7HMR2 136264453 IC50 = 37 nM T39231 CUPY84 136268378 IC50 = 65.4 nM T39231 CF3X4M 136372378 IC50 = 101 nM T39231 CUB67C 136404917 IC50 > 100000 nM T39231 CWH02F 136491252 IC50 = 47 nM T39231 CF80AR 136491263 IC50 = 111 nM T39231 C6T9OI 136947736 IC50 = 2.2 nM T39231 C91WJF 136947741 IC50 = 1.3 nM T39231 CFS5Z4 136947743 IC50 = 31 nM T39231 CVM4S9 136947751 IC50 = 35 nM T39231 C9UGV5 137169064 IC50 = 19.4 nM T39231 CMN5H6 137169065 IC50 = 21.3 nM T39231 CF8LC7 137632525 IC50 = 977.24 nM T39231 C8K3CX 137634198 IC50 = 31.62 nM T39231 CS7ZQ8 137637696 IC50 = 33.88 nM T39231 C7V2RQ 137640411 IC50 = 7943.28 nM T39231 CJE2O1 137642565 IC50 = 2691.53 nM T39231 C46GFQ 137643877 IC50 = 6000 nM T39231 CM21PL 137646367 IC50 = 575.44 nM T39231 CIF2B4 137646395 IC50 = 10000 nM T39231 C34NWB 137649146 IC50 = 158.49 nM T39231 CG0P8H 137650831 IC50 = 9332.54 nM T39231 CD0E9C 137653685 IC50 > 10000 nM T39231 C5ZX2H 137653831 IC50 = 7943.28 nM T39231 CX2HY9 137656402 IC50 > 10000 nM T39231 C4UTR7 137656957 IC50 = 4786.3 nM T39231 C72FHM 137660379 IC50 = 9772.37 nM T39231 C74JDS 137660681 IC50 = 1.995 nM T39231 C4R7VI 137701512 IC50 = 14.3 nM T39231 CWLV03 138594154 IC50 = 7.9 nM T39231 CDW5N1 138594164 IC50 = 4.9 nM T39231 CSK82I 138594166 IC50 = 4.8 nM T39231 CD1M0Y 138594171 IC50 = 12.8 nM T39231 C9QYJ3 138594172 IC50 = 11.1 nM T39231 C1XSH7 138594194 IC50 = 36.1 nM T39231 C4JO9N 138594198 IC50 = 3.7 nM T39231 C7I1CT 138594235 IC50 = 13.6 nM T39231 CVI5N9 138594242 IC50 = 7.5 nM T39231 CS8U3T 138594273 IC50 = 9.2 nM T39231 CYR32Z 138594277 IC50 = 3.8 nM T39231 CNSV30 138594278 IC50 = 6.1 nM T39231 C1C2AS 138594290 IC50 = 12 nM T39231 C34OCY 138594292 IC50 = 5.5 nM T39231 CUA1E8 138594320 IC50 = 3.5 nM T39231 CGE6Q5 138594327 IC50 = 11.1 nM T39231 C0RST4 138594360 IC50 = 33.7 nM T39231 C4K7MW 138594363 IC50 = 4.4 nM T39231 CNW2O9 138594369 IC50 = 6.4 nM T39231 C3F7MV 138594378 IC50 = 7.5 nM T39231 C6YU8S 138594385 IC50 = 16 nM T39231 C48AGS 138594414 IC50 = 28.5 nM T39231 CA49EZ 138594436 IC50 = 43.4 nM T39231 CL6EV4 138594465 IC50 = 4.2 nM T39231 CJL05F 138594467 IC50 = 9.9 nM T39231 CX4SL6 138594472 IC50 = 4.4 nM T39231 C3E5IU 138594491 IC50 = 14.1 nM T39231 C13EVQ 138594498 IC50 = 31.5 nM T39231 C4L9XQ 138594506 IC50 = 49.3 nM T39231 CKF1W3 138594528 IC50 = 11.1 nM T39231 C98NUR 138594556 IC50 = 4.4 nM T39231 CDZ43N 138594558 IC50 = 7.9 nM T39231 CLD3J5 138594570 IC50 = 7.7 nM T39231 CWVO67 138594578 IC50 = 18.2 nM T39231 C6QD2W 138594607 IC50 = 10.2 nM T39231 CP6Y5L 138594610 IC50 = 4.5 nM T39231 CSQJ12 138594627 IC50 = 5.3 nM T39231 CEOJ61 138594628 IC50 = 5.8 nM T39231 CU4O9K 138594631 IC50 = 5.3 nM T39231 C0A4FG 138594645 IC50 = 11 nM T39231 CN3U9X 138594667 IC50 = 9 nM T39231 CQK29G 138594732 IC50 = 8.4 nM T39231 CCU4I1 138594747 IC50 = 6.4 nM T39231 C1KWY7 138594763 IC50 = 5.8 nM T39231 C9HR2J 138594785 IC50 = 30.2 nM T39231 CP4NF9 138594790 IC50 = 27.6 nM T39231 CF74SW 138594809 IC50 = 16.8 nM T39231 CF7ZR5 138594952 IC50 = 10 nM T39231 CW5E6D 138594964 IC50 = 16.7 nM T39231 CURM89 138594969 IC50 = 16.6 nM T39231 C72QVS 138595093 IC50 = 118 nM T39231 C8I9CD 142613964 IC50 = 5.4 nM T39231 C5SG1U 145957836 IC50 = 1000 nM T39231 CPR0N4 145962722 IC50 > 100000 nM T39231 C6HOA3 145972257 IC50 = 5700 nM T39231 CA65UC 145974539 IC50 = 3000 nM T39231 C20TJH 145987470 IC50 = 11000 nM T39231 COB76P 145989667 IC50 = 131 nM T39231 CPY72O 153951026 IC50 = 15 nM T39231 CWV08R 155511996 IC50 = 1350 nM T39231 CZ78CA 155513337 IC50 = 14300 nM T39231 CRX36I 155515281 IC50 = 4.3 nM T39231 CC9J2N 155516254 IC50 = 6.3 nM T39231 C6EJ7I 155518170 IC50 = 7779 nM T39231 CIC9H8 155518184 IC50 = 14.9 nM T39231 C1DL6E 155518640 IC50 = 220 nM T39231 CGKW04 155520067 IC50 > 20000 nM T39231 CHV6T4 155521523 IC50 = 2.5 nM T39231 CUM52X 155522687 IC50 = 3.4 nM T39231 CEP6Y5 155528458 IC50 = 79.6 nM T39231 C91IPT 155529963 IC50 = 8.9 nM T39231 CA9XP1 155531429 IC50 = 28.5 nM T39231 CL2PO4 155532179 IC50 = 10.3 nM T39231 C09PYD 155532212 IC50 = 67.6 nM T39231 C4JPD1 155532717 IC50 = 21.3 nM T39231 CZL4U1 155534087 IC50 = 16.2 nM T39231 CV2MX1 155535415 IC50 = 35 nM T39231 CY8RJ7 155537249 IC50 = 131 nM T39231 CWM48X 155538013 IC50 = 19.4 nM T39231 CU65VW 155540828 IC50 = 514 nM T39231 CZN0O1 155541146 IC50 = 5919 nM T39231 CYWG48 155541643 IC50 > 1000 nM T39231 C9INM1 155543325 IC50 = 9.2 nM T39231 CG0J7F 155545779 IC50 = 6.3 nM T39231 CO0E8F 155549220 IC50 = 6.2 nM T39231 CD5C9R 155550189 IC50 > 20000 nM T39231 C4P3QD 155553178 IC50 = 19 nM T39231 CIYH06 155556919 IC50 = 6168 nM T39231 CXAJ25 155557028 IC50 = 53.5 nM T39231 CWH8D0 155561438 IC50 = 7.8 nM T39231 C46UYI 155562058 IC50 = 6008 nM T39231 COH6X1 155564702 IC50 = 6.8 nM T39231 D00RIX 5280443 IC50 = 3162.28 nM T39231 D00TUB 135471356 IC50 = 83 nM T39231 D02CHG 248021 IC50 = 588.84 nM T39231 D03BQJ 688829 IC50 = 47 nM T39231 D04GFX 736736 IC50 > 10000 nM T39231 D04WDX 4858 IC50 = 1348.96 nM T39231 D06NKJ 135439437 IC50 = 475 nM T39231 D07BPT 135457978 IC50 = 32 nM T39231 D0B2WX 135407310 IC50 = 37 nM T39231 D0C5XB 261395 IC50 = 208.93 nM T39231 D0E5EW 135531482 IC50 = 42 nM T39231 D0G5VD 135492389 IC50 = 58 nM T39231 D0GA0Y 135463623 IC50 = 35 nM T39231 D0O6WW 135528341 IC50 = 195 nM T39231 D0OF1I 135417274 IC50 = 873 nM T39231 D0P3CX 689013 IC50 > 10000 nM T39231 D0S0RK 10680 IC50 = 323.59 nM T39231 D0Y1MH 135471354 IC50 = 52 nM T39231 D0YJ3Q 5322065 IC50 = 630 nM T34287 CQ2B5Z 44313403 IC50 = 140000 nM T34287 CH7W9F 44313519 IC50 = 39000 nM T34287 CFEN62 44313520 IC50 = 40000 nM T34287 CQWZ67 44313524 IC50 = 34000 nM T34287 CD2O9V 44313525 IC50 > 200000 nM T34287 CHGO46 44313559 IC50 > 200000 nM T34287 C7GEA5 44313560 IC50 > 200000 nM T34287 CXN3V4 44313599 IC50 = 50000 nM T34287 CLIX86 44313609 IC50 = 14000 nM T34287 CXG87J 44313676 IC50 = 34000 nM T34287 CCP04F 44313751 IC50 > 200000 nM T34287 C0CD4S 44313774 IC50 > 200000 nM T34287 C74CAN 44313775 IC50 = 93000 nM T34287 CYQU68 44313793 IC50 = 21000 nM T34287 CL81DH 44313818 IC50 = 50000 nM T34287 C2BL4S 44313832 IC50 = 15000 nM T34287 C0C7MZ 44313842 IC50 = 6000 nM T34287 CMJ68T 44313861 IC50 > 200000 nM T34287 CCUH40 44313876 IC50 > 200000 nM T34287 C75VKP 44313877 IC50 > 200000 nM T34287 CIVW97 44313898 IC50 > 500000 nM T34287 CYRQ36 44314130 IC50 = 30000 nM T76396 C8SGZ7 9799609 IC50 > 20000 nM T76396 C2H4ZK 9806118 IC50 = 12000 nM T76396 C2TN7S 9807068 IC50 > 50000 nM T76396 C71XRT 9821510 IC50 = 40000 nM T76396 CEL3C9 9824630 IC50 > 50000 nM T76396 CXE1Y8 9842436 IC50 > 20000 nM T76396 CISP20 9844227 IC50 = 11000 nM T76396 CNE6P0 9845017 IC50 = 11000 nM T76396 C7VSU2 9845018 IC50 = 3400 nM T76396 CXH80T 9845019 IC50 = 15000 nM T76396 CNIS42 9846821 IC50 = 24 nM T76396 CML5U3 9848397 IC50 = 15000 nM T76396 CXZ6Q7 9866918 IC50 > 20000 nM T76396 C0QV1K 9871743 IC50 = 12000 nM T76396 C4NJS0 9885760 IC50 = 41000 nM T76396 CRW8C1 9907452 IC50 = 46000 nM T76396 CA8KC0 9912881 IC50 > 50000 nM T76396 CW1KP6 9914569 IC50 = 4600 nM T76396 CF85LV 9915185 IC50 = 6500 nM T76396 CH2KA7 9930818 IC50 = 48000 nM T76396 CY7W8H 9931146 IC50 = 42000 nM T76396 CI8P9X 9952087 IC50 = 46000 nM T76396 CNRX39 9956928 IC50 = 1100 nM T76396 CT3O4V 10138186 IC50 = 4800 nM T76396 CNET60 10206356 IC50 = 1100 nM T76396 C5BJ0E 10238214 IC50 = 3900 nM T76396 COJI94 10862667 IC50 > 50000 nM T76396 C3SM0F 10894628 IC50 = 7400 nM T76396 C4QZ2E 10895064 IC50 = 11000 nM T76396 C5L2FR 10896860 IC50 = 3600 nM T76396 C3T9CI 10916025 IC50 = 16000 nM T76396 C3SQA5 10918896 IC50 = 2700 nM T76396 CYJ0H9 10938254 IC50 > 50000 nM T76396 CG34TZ 10949393 IC50 > 50000 nM T76396 CR8NL2 10950878 IC50 > 50000 nM T76396 C7MJ3I 10960344 IC50 = 11000 nM T76396 CL3A7F 10961614 IC50 = 41000 nM T76396 CS1CI9 10982914 IC50 = 28000 nM T76396 CIS36R 10993420 IC50 > 50000 nM T76396 CJI01L 11004204 IC50 = 1500 nM T76396 C2BX4N 11025461 IC50 = 24000 nM T76396 CPXY41 11037188 IC50 = 19000 nM T76396 CKZP84 11048052 IC50 = 19000 nM T76396 CR9K5V 11069519 IC50 = 6500 nM T76396 CN6QM7 11080796 IC50 ~ 5100 nM T76396 CV73YG 11091386 IC50 = 880 nM T76396 CBY94W 11091976 IC50 = 20000 nM T76396 CY0F2S 11101410 IC50 = 31000 nM T76396 C9COS1 11101729 IC50 = 2800 nM T76396 CRL01V 11111808 IC50 = 14000 nM T76396 CUT1Q0 11728765 IC50 > 50000 nM T76396 C30TBM 11732162 IC50 > 50000 nM T76396 CA4I7V 11824866 IC50 = 36000 nM T76396 C80JFP 17965976 IC50 = 100 nM T76396 C74LVI 44274781 IC50 = 10 nM T76396 C34TGF 44274782 IC50 = 5600 nM T76396 C4XQY2 44274783 IC50 = 1200 nM T76396 C2PNA5 44274804 IC50 = 210 nM T76396 C2U0NZ 44274806 IC50 = 240 nM T76396 CA9MJ4 44274825 IC50 = 1800 nM T76396 CM12CG 44286282 IC50 = 650 nM T76396 C5W8QG 44286298 IC50 = 2800 nM T76396 C4O9EB 44286300 IC50 = 4200 nM T76396 CGOQ58 44286304 IC50 = 2600 nM T76396 CI67NQ 44286315 IC50 = 2100 nM T76396 C2U6PY 44286332 IC50 = 3900 nM T76396 C9QSC5 44286345 IC50 = 2400 nM T76396 C9BH3L 44286376 IC50 = 1200 nM T76396 C5Y8HE 44286420 IC50 = 510 nM T76396 C08IJY 44286579 IC50 = 1600 nM T76396 CT1QP4 44286646 IC50 > 10 nM T76396 CWSA69 44286656 IC50 > 10 nM T76396 C5NG4A 44286723 IC50 = 1100 nM T76396 C4E1KL 44286730 IC50 = 5500 nM T76396 CFO4S0 44286731 IC50 > 10 nM T76396 CCD43U 44286732 IC50 = 42 nM T76396 CQH1L4 44286733 IC50 = 1400 nM T76396 CAH5P4 44286737 IC50 > 10 nM T76396 CENW21 44286755 IC50 = 830 nM T76396 C2I9BP 44286765 IC50 = 1700 nM T76396 C7XLA6 44286767 IC50 > 10 nM T76396 C05LZF 44286768 IC50 = 2100 nM T76396 CYS6L1 44286776 IC50 = 103 nM T76396 C8QG1O 44286780 IC50 = 1800 nM T76396 CKH50S 44286801 IC50 = 990 nM T76396 CT46KR 44286802 IC50 = 8620 nM T76396 CW64TF 44286942 IC50 > 10 nM T76396 CLPC20 44286957 IC50 = 960 nM T76396 C0S4NX 44286958 IC50 > 10 nM T76396 C42IDV 44286959 IC50 = 8600 nM T76396 CNO31Q 44459100 IC50 = 18 nM T76396 CI9ZK4 44459321 IC50 = 40 nM T76396 CN02QA 44459344 IC50 = 740 nM T76396 COA1V2 44459504 IC50 = 430 nM T76396 CEJ0K9 44459509 IC50 = 4100 nM T76396 CL8G5A 44459510 IC50 = 870 nM T76396 CAD74Y 44459594 IC50 = 2400 nM T76396 CG4LH7 44459775 IC50 = 3.1 nM T76396 C39TIB 44459799 IC50 = 360 nM T76396 C6RBS7 44459800 IC50 = 83000 nM T76396 C97BTH 44459819 IC50 = 9.5 nM T76396 CF2XW7 44459847 IC50 = 16 nM T76396 C4KA0M 44459853 IC50 = 92 nM T76396 C7V4FJ 44459924 IC50 > 10000 nM T93788 D00WDY 53477157 EC50 = 14 nM T93788 D01HTO 25025505 EC50 = 87 nM T93788 D0O9XN 11691484 EC50 = 46 nM T93788 D0S4II 24996872 EC50 = 3.4 nM T93788 D0Q3ES 11705608 EC50 = 2.7 nM T93788 C1JLP6 1267327 EC50 = 310 nM T93788 C12OPB 3710394 EC50 = 1000 nM T93788 CT6HM1 3766553 IC50 = 84 nM T93788 CL19MX 3800660 EC50 = 3000 nM T93788 CW7I0V 4400062 EC50 = 200 nM T93788 CBM61L 4993934 EC50 = 1900 nM T93788 C09VLS 10003301 EC50 = 2500 nM T93788 C0VR7W 10049468 IC50 = 50 nM T93788 C14WGV 10094886 EC50 = 1700 nM T93788 C43IKO 11190983 EC50 = 15 nM T93788 CPN90M 11224944 EC50 = 3.5 nM T93788 CA50RX 11271133 EC50 = 14 nM T93788 C7T4LO 11271424 EC50 = 4.2 nM T93788 CM7CW0 11283457 EC50 = 116 nM T93788 CCO2Y6 11397354 EC50 = 0.7 nM T93788 CL4J5R 11465648 EC50 = 7.4 nM T93788 CR5I6K 11503692 EC50 = 9.7 nM T93788 C5GVB6 11641004 EC50 = 31 nM T93788 CS3RW4 11663249 EC50 = 44 nM T93788 C2QWX4 11677830 EC50 = 71 nM T93788 CB4XD1 11691227 EC50 = 1320 nM T93788 C2T8FN 11751802 EC50 = 250 nM T93788 CO36JD 16036825 EC50 = 7.3 nM T93788 CA7P1J 16733804 EC50 = 200 nM T93788 CO8BD9 21897416 EC50 > 10000 nM T93788 COMA70 21897603 EC50 = 2400 nM T93788 C6ARZ3 21897616 EC50 = 435 nM T93788 CDM28O 21897675 EC50 = 8.1 nM T93788 C93QDC 21897744 EC50 = 50.12 nM T93788 CGH9P2 21897819 EC50 > 10000 nM T93788 CACM74 21897825 EC50 = 316.23 nM T93788 C2OVZ5 21897897 EC50 = 5.6 nM T93788 CR0VF4 23649212 EC50 = 131 nM T93788 CBZF78 23653563 EC50 = 50.12 nM T93788 CR9J5G 24822706 EC50 = 22 nM T93788 CE0UN4 24862850 EC50 = 400 nM T93788 C4YU8M 24896777 EC50 = 251.19 nM T93788 C0IXZ8 24896778 EC50 = 10 nM T93788 C06AXF 24897005 EC50 = 19.95 nM T93788 CZJ7U6 24897242 EC50 = 125.89 nM T93788 CXGZ83 24897245 EC50 > 10000 nM T93788 CLNB23 24897458 EC50 = 316.23 nM T93788 CJ9F7N 24897459 EC50 = 251.19 nM T93788 CR04JD 24897884 EC50 > 10000 nM T93788 CML3Z6 24897885 EC50 = 794.33 nM T93788 CLS39J 24898315 EC50 = 1995.26 nM T93788 CHRG37 24899742 EC50 = 12.59 nM T93788 C68CJU 24899747 EC50 = 1584.89 nM T93788 CFD7Y9 24899748 EC50 = 1258.93 nM T93788 CT9OL3 24899996 EC50 = 398.11 nM T93788 C89JDC 24900242 EC50 > 10000 nM T93788 CXF35U 24900244 EC50 = 31.62 nM T93788 C7I8XM 24958871 EC50 = 25 nM T93788 C04VLG 24958872 EC50 = 338 nM T93788 C3QYJ8 24961071 EC50 = 514 nM T93788 C8ZYQ0 24961798 EC50 = 6 nM T93788 CKT12U 24961799 EC50 = 6 nM T93788 CHI91S 24961800 EC50 = 1 nM T93788 CCK8G4 25012362 EC50 = 8 nM T93788 CU72GZ 25012522 EC50 = 98 nM T93788 C0EI7T 25012524 EC50 = 2 nM T93788 C85YLN 25012528 EC50 = 201 nM T93788 CO7AD3 25024141 EC50 = 103 nM T93788 CN75ZE 25052772 EC50 = 19 nM T93788 CP7NC9 25052969 IC50 = 500 nM T93788 C06OMU 25052970 EC50 = 1200 nM T93788 CVF60B 25053040 EC50 = 400 nM T93788 COHV79 25053041 EC50 = 260 nM T93788 C6TQH7 25053042 EC50 = 10 nM T93788 CB9EU8 25053043 EC50 = 430 nM T93788 CN9O5M 25053044 EC50 = 25 nM T93788 C16MFX 25053111 EC50 = 160 nM T93788 C49GZF 25053112 EC50 = 5.1 nM T93788 C85TLK 25053113 EC50 = 1.5 nM T93788 C7E1UM 25053114 EC50 = 660 nM T93788 C9C1PY 25053115 EC50 = 24 nM T93788 C5E0RZ 25053184 EC50 = 17 nM T93788 C0NSW2 25053185 EC50 = 4.7 nM T93788 C8JVE4 25053186 EC50 = 7.8 nM T93788 CN1KA0 25053187 EC50 = 17.1 nM T93788 CY6G1Q 25053188 EC50 = 110 nM T93788 CESK31 25053253 EC50 = 3.4 nM T93788 CM3OE2 25053254 EC50 = 7 nM T93788 CX73WG 25053255 EC50 = 7.9 nM T93788 CZNB62 25138357 EC50 = 133 nM T93788 CMT76B 25138367 EC50 = 63 nM T93788 CS2K9L 25204037 EC50 = 23 nM T93788 C0V6PX 25204038 EC50 = 16 nM T93788 CCO6Y1 25204174 EC50 = 183 nM T93788 C2GC5X 25204242 EC50 = 1700 nM T93788 CG5DU7 25204244 EC50 = 1091 nM T93788 C50QKG 25204645 EC50 = 57 nM T93788 C8GQY7 25204648 EC50 = 724 nM T93788 C9X8DN 25204713 EC50 = 130 nM T93788 C4FIJ0 25260830 EC50 = 17 nM T93788 CYOT98 42646474 EC50 = 95 nM T93788 CO9R2B 44177589 EC50 = 39.81 nM T93788 CMD02U 44177592 EC50 = 794.33 nM T93788 C82IAU 44177593 EC50 > 10000 nM T93788 C8WM0Z 44467183 EC50 = 2 nM T93788 C5ETU8 44467185 EC50 = 4 nM T93788 CYU89I 46208490 Ki = 20 nM T93788 CGI81S 46865202 EC50 = 90 nM T93788 CK42WB 46865203 EC50 = 300 nM T93788 C91WPT 46884780 EC50 > 10000 nM T93788 C4I0MC 46884781 EC50 > 10000 nM T93788 CDTI38 46884819 EC50 > 10000 nM T93788 CZ1QG5 46884820 EC50 = 1900 nM T93788 CND62Y 46884821 EC50 = 2600 nM T93788 CMIP79 46884822 EC50 = 1300 nM T93788 CEGR15 46884857 EC50 = 300 nM T93788 CF2SO1 46884858 EC50 = 100 nM T93788 CJ45TU 46884859 EC50 = 300 nM T93788 CU5KI2 46884902 EC50 = 200 nM T93788 CQDL72 46884903 EC50 = 2000 nM T93788 CB0L3Y 46884904 EC50 = 1800 nM T93788 CS4RO2 46884935 EC50 = 1200 nM T93788 CS1U6Z 46884936 EC50 = 1000 nM T93788 CTY74I 46884937 EC50 = 1000 nM T93788 CNDH97 46884938 EC50 = 1600 nM T93788 C3MZY2 46884986 EC50 = 800 nM T93788 CF8T7O 46884987 EC50 = 2800 nM T93788 C2CIG9 46884988 EC50 > 10000 nM T93788 C1V4KW 46884989 EC50 = 2100 nM T93788 CE71WG 46885048 EC50 = 2000 nM T93788 CVIS54 46885049 EC50 > 10000 nM T93788 CK9TR7 46885050 EC50 = 900 nM T93788 C5JNL7 46885051 EC50 = 2100 nM T93788 C0YZ8U 46885169 EC50 = 1200 nM T93788 COPL82 46885170 EC50 = 700 nM T93788 CIH1K7 46885171 EC50 = 130 nM T93788 C2H5OS 46897575 EC50 = 7.7 nM T93788 CF7UP1 46897577 EC50 = 11 nM T93788 CIF0Y7 46939910 EC50 = 15 nM T93788 C9L4ZU 49855246 EC50 = 1 nM T93788 CC27AL 51029601 EC50 = 65 nM T93788 CWJ36V 51029603 EC50 = 621 nM T93788 CSW80J 51029782 EC50 = 1925 nM T93788 CW19DN 51029876 IC50 = 17 nM T93788 CXJ30Q 51029877 EC50 = 466 nM T93788 CBR8Z2 51029964 EC50 = 45 nM T93788 CPYT82 51029965 EC50 = 3 nM T93788 CY0B7Q 51030053 EC50 = 21 nM T93788 CM0UF3 51030054 EC50 = 5 nM T93788 CW08DZ 51030056 EC50 = 63 nM T93788 C5LO4C 51030336 EC50 = 112 nM T93788 CVY9U0 51030529 EC50 = 54 nM T93788 C07HID 51030707 EC50 = 630.96 nM T93788 CM9PY8 51030710 IC50 = 12 nM T93788 CP6NI2 51030711 EC50 = 7.943 nM T93788 CTI6N7 51030811 EC50 = 75 nM T93788 CZLP32 51030896 EC50 = 21 nM T93788 C1P9UY 51030897 EC50 = 5 nM T93788 CW06HL 51030898 EC50 = 10 nM T93788 C9D8FG 51030899 EC50 = 15.85 nM T93788 CS4X5Z 51030900 EC50 = 15.85 nM T93788 C4QW2B 51030901 EC50 = 2 nM T93788 C70OGS 51030984 EC50 = 20 nM T93788 CX28ZP 51030985 EC50 = 47 nM T93788 C9W8OF 51030987 EC50 = 14 nM T93788 C35XAI 51354342 EC50 = 740 nM T93788 CBG8N3 51354343 EC50 = 2067 nM T93788 C2RCZ0 53235503 EC50 = 3 nM T93788 C6OJF7 53317209 EC50 = 267 nM T93788 CR06WM 53317210 EC50 = 340 nM T93788 C2O9SZ 53317211 EC50 = 868 nM T93788 CT2D0R 53318456 EC50 = 884 nM T93788 CQ8GY0 53318501 EC50 = 808 nM T93788 CV8P3R 53318502 EC50 = 32 nM T93788 C0S9BL 53319831 EC50 = 1380 nM T93788 C0I8YS 53321124 EC50 = 120 nM T93788 CO1HB3 53322450 EC50 = 78 nM T93788 C85UDG 53322927 EC50 = 5980 nM T93788 CO98ZY 53323811 EC50 = 75 nM T93788 CIBE50 53325083 EC50 = 409 nM T93788 CUJ28D 53326341 EC50 = 13 nM T93788 C49ZMH 53390936 EC50 = 13 nM T93788 CHN72W 53469852 EC50 = 4 nM T93788 CP4AU5 53477048 EC50 = 13 nM T93788 CFT8B9 53477049 EC50 = 12 nM T93788 C5I8FB 53477155 EC50 = 16 nM T93788 CXE8V4 53477156 EC50 = 18 nM T93788 CO4S6E 53491642 EC50 = 8.6 nM T93788 C8XHK5 53491715 EC50 = 25.9 nM T93788 C3BFK2 53491780 EC50 = 65.1 nM T93788 C5HV3A 53491781 EC50 = 18.5 nM T93788 C8K0CB 53491782 EC50 = 31.1 nM T93788 C4OC7H 53492264 EC50 = 4.8 nM T93788 C16SZL 53492331 EC50 = 1.2 nM T93788 CGE8C9 53492397 EC50 = 62.6 nM T93788 CCE83O 53492463 EC50 = 54.8 nM T93788 CDQ2M4 53492467 EC50 = 16.1 nM T93788 CQK96E 53492528 EC50 = 8.5 nM T93788 CUJ76Z 53492593 EC50 = 262 nM T93788 C08XHA 53492594 EC50 = 5.9 nM T93788 CQUT71 53630395 EC50 = 11.6 nM T93788 C9K5GR 53630396 EC50 = 265 nM T93788 C1J8XI 53630398 EC50 = 6.3 nM T93788 C9M4QV 53630415 EC50 = 3.8 nM T93788 CEA18U 53630423 EC50 = 33.4 nM T93788 CRS4L7 53630450 EC50 = 14.6 nM T93788 C7EQT9 54580684 EC50 = 2580 nM T93788 CQWV19 54580747 EC50 = 5 nM T93788 C17ICO 54580903 EC50 = 526 nM T93788 CTJA61 54580904 EC50 = 48 nM T93788 C20FZY 54581118 EC50 = 3.4 nM T93788 C3IP1A 54581957 EC50 = 1400 nM T93788 CA37UQ 54581959 EC50 = 103 nM T93788 CDW8U1 54581961 EC50 = 62 nM T93788 C8CTD7 54581962 EC50 = 9 nM T93788 C7APK5 54582694 EC50 = 1150 nM T93788 CZ71VB 54582892 EC50 = 0.2 nM T93788 CZ6KG9 54583401 EC50 = 1239 nM T93788 CQ70UX 54583648 EC50 = 860 nM T93788 CCN3K0 54583892 EC50 = 600 nM T93788 C7GMD0 54583893 EC50 = 39 nM T93788 CL24JP 54583894 EC50 = 57 nM T93788 CG78OW 54583895 EC50 = 30 nM T93788 CSCE48 54583896 EC50 = 20 nM T93788 CY05QH 54584353 Ki = 20 nM T93788 CM1JT0 54584624 EC50 > 20000 nM T93788 CWBJ19 54584625 EC50 = 82 nM T93788 CL8MW9 54584841 EC50 = 76 nM T93788 CIVJ34 54585040 EC50 = 3.4 nM T93788 CR2OQ6 54585806 EC50 = 1900 nM T93788 CDK61R 54585807 EC50 = 11 nM T93788 CS2J3H 54585808 EC50 = 18 nM T93788 C3H6IN 54585809 EC50 = 13 nM T93788 CY4FD8 54586012 EC50 = 42 nM T93788 C64MJP 54586548 EC50 = 558 nM T93788 CEL6P0 54586563 EC50 = 130 nM T93788 CUZF70 54586564 EC50 = 918 nM T93788 C5CGF7 54586777 EC50 = 116 nM T93788 CK5ZC4 54586778 EC50 = 2 nM T93788 C6KS2N 54586779 EC50 = 19 nM T93788 C67NFK 54586780 EC50 = 19 nM T93788 C4ACJ8 54586781 EC50 = 2 nM T93788 CPO85I 54586882 EC50 = 7.5 nM T93788 C03XYL 54586987 EC50 = 7.3 nM T93788 CK3D9N 54587592 EC50 = 62 nM T93788 C39VDT 54587812 EC50 = 831 nM T93788 CZ5IY9 54587813 EC50 = 0.3 nM T93788 C1WZ4V 54589149 EC50 = 60 nM T93788 CO3C4B 54589151 EC50 = 62 nM T93788 C49WCU 54589190 EC50 = 544 nM T93788 CIYV57 54589191 EC50 = 1003 nM T93788 CO7F6Q 54589229 EC50 = 521 nM T93788 C73SNB 54589230 EC50 = 14 nM T93788 C2SNJ3 54589231 EC50 = 78 nM T93788 C8L1JO 54589232 EC50 = 51 nM T93788 C54UCK 54589269 EC50 = 16 nM T93788 C2SP3B 54589270 EC50 = 101 nM T93788 COJI15 54596144 EC50 = 13.7 nM T93788 C7QB1F 56591900 EC50 = 129 nM T93788 CKN41C 56592326 EC50 = 53 nM T93788 C2YXS6 56592327 EC50 = 41 nM T93788 CB2I9X 56592328 EC50 = 42 nM T93788 CF46NB 56592329 EC50 = 79 nM T93788 CMZ0G6 56592412 EC50 > 1000 nM T93788 CM0IL4 56592414 EC50 > 1000 nM T93788 CM1DB2 56592599 EC50 > 1000 nM T93788 C9ZF6B 56643412 EC50 = 74 nM T93788 C0MQ2W 56832511 EC50 = 24 nM T93788 CKC63L 56943106 EC50 = 23.4 nM T93788 C21XMN 56961034 EC50 = 353 nM T93788 C91JWV 56963355 EC50 = 27 nM T93788 CB5V4R 56963356 EC50 = 28.2 nM T93788 C3EL1T 57390603 EC50 = 260 nM T93788 C1C5TR 57390604 EC50 = 2330 nM T93788 CMF49J 57392378 EC50 = 235 nM T93788 CXL42B 57392379 EC50 = 60 nM T93788 CC75BU 57392380 EC50 = 60 nM T93788 C5E9UK 57392504 EC50 = 47 nM T93788 CZKU95 57393406 EC50 = 1410 nM T93788 COHW15 57394106 EC50 = 1000 nM T93788 C2A4UT 57394950 EC50 = 120 nM T93788 CBDV65 57397673 EC50 = 92 nM T93788 CWX87F 57397674 EC50 = 490 nM T93788 CU6O0S 57397675 EC50 = 210 nM T93788 CL0XS2 57397676 EC50 = 132 nM T93788 C8DJ9M 57399342 EC50 = 34 nM T93788 C89CRJ 57399343 EC50 > 5000 nM T93788 C4GXR6 57399344 EC50 = 25 nM T93788 C7HKF8 57399345 EC50 > 5000 nM T93788 CH6KB4 57401105 EC50 = 475 nM T93788 CI1SJ3 57401106 EC50 = 250 nM T93788 C6QIP7 57401198 EC50 = 1100 nM T93788 CBZ4C3 57402128 EC50 = 5.4 nM T93788 CD68KC 57402865 EC50 = 50 nM T93788 C7AGB4 57403665 EC50 = 115 nM T93788 C08QUG 57404926 EC50 = 3423 nM T93788 CYO3V8 57405092 EC50 = 14 nM T93788 CS5P8Y 57415237 EC50 = 100 nM T93788 C1TDX7 57468373 EC50 = 104 nM T93788 C7D5BO 57468382 EC50 = 117 nM T93788 CGI92M 57468398 EC50 = 31 nM T93788 CD7SN3 57468401 EC50 > 10000 nM T93788 C7T2OX 57468409 EC50 = 9 nM T93788 CFA0K6 57468427 EC50 = 5 nM T93788 CYX6F2 57468435 EC50 = 32 nM T93788 C12DVB 57468459 EC50 = 11 nM T93788 C7VF2J 57550042 EC50 = 18 nM T93788 CI63JT 57550050 EC50 = 870 nM T93788 CN4AZ7 57550070 EC50 = 41 nM T93788 C3ANB4 57550087 EC50 = 37 nM T93788 CGAF21 57550101 EC50 = 12 nM T93788 CT4XG6 58016984 EC50 = 79.43 nM T93788 C8Z2EV 58016989 EC50 = 50.12 nM T93788 CSX9K6 58016997 EC50 > 10000 nM T93788 C91ITW 58016999 EC50 = 630.96 nM T93788 CN4B6V 58017000 EC50 = 158.49 nM T93788 CS0B5T 58017005 EC50 = 316.23 nM T93788 CH1IX9 58017008 EC50 = 1995.26 nM T93788 CR3NF9 58017011 EC50 = 79.43 nM T93788 CE15RN 58017018 EC50 = 125.89 nM T93788 CPJD17 58017023 EC50 = 501.19 nM T93788 CSQ59A 58017025 EC50 = 100 nM T93788 CS7JH1 58017027 EC50 = 501.19 nM T93788 CTIP85 58017028 EC50 = 125.89 nM T93788 CX61OG 58017032 EC50 = 79.43 nM T93788 CZ2QA6 58017033 EC50 = 25.12 nM T93788 CU63JN 58017035 EC50 = 251.19 nM T93788 C9W8VD 58017036 EC50 = 79.43 nM T93788 C32MKS 58017038 EC50 = 158.49 nM T93788 CZE6U9 58017039 EC50 = 251.19 nM T93788 C84HGI 58017045 EC50 = 63.1 nM T93788 CZHW78 58017047 EC50 = 1000 nM T93788 CF86HB 58017059 EC50 = 398.11 nM T93788 C2LP9G 58074082 EC50 = 16 nM T93788 CKCV24 58114293 EC50 = 43.6 nM T93788 CO95HL 58116587 EC50 = 87 nM T93788 CDY74O 58116595 EC50 = 8800 nM T93788 C6L8YG 58190314 EC50 = 6 nM T93788 CH64EP 58190317 EC50 = 19.95 nM T93788 C7AY1J 58190324 EC50 = 12 nM T93788 C10KEY 58190329 EC50 = 63.1 nM T93788 CI63UA 58190330 EC50 = 20 nM T93788 CAGF43 58190343 EC50 = 64 nM T93788 C2L8TG 58190347 EC50 = 54 nM T93788 C3A4KQ 58190389 EC50 = 39 nM T93788 C5K1EG 58190395 EC50 = 2217 nM T93788 CA4G8T 58190401 EC50 = 234 nM T93788 C3PA2V 58190405 EC50 = 41 nM T93788 CON8B6 58190423 EC50 = 54 nM T93788 CB0V9M 59234074 EC50 = 353 nM T93788 CC1L3O 60152410 EC50 = 31 nM T93788 C5NW9S 60155096 EC50 = 1084 nM T93788 C0Z1NG 60155097 EC50 = 485 nM T93788 C84NFQ 60155098 EC50 > 30000 nM T93788 CHN8K5 60155099 EC50 = 186 nM T93788 C4YBX8 60155100 EC50 = 737 nM T93788 CQ34SH 60155182 EC50 > 7500 nM T93788 CU69NX 60155183 EC50 = 161 nM T93788 C7RYQ5 60155184 EC50 = 893 nM T93788 CI28PS 60155273 EC50 = 156 nM T93788 CXP75O 60155274 EC50 = 29 nM T93788 C9LGW7 60155364 EC50 = 79 nM T93788 C5F3JO 60155365 EC50 = 39 nM T93788 C4VJ1C 60155366 EC50 = 16 nM T93788 C18HZU 60155367 EC50 > 1937 nM T93788 CXA1Q4 60155457 EC50 = 63 nM T93788 CM3OX4 60155458 EC50 > 30000000 nM T93788 CG03LC 60155459 EC50 = 154 nM T93788 C6XG4H 60155460 EC50 = 184 nM T93788 C4TH9X 60155461 EC50 = 100 nM T93788 CL41YN 60155543 EC50 = 25 nM T93788 CX0PT7 62706030 EC50 = 51 nM T93788 CPR29D 62706192 EC50 = 210 nM T93788 CBR1J6 62706193 EC50 = 145 nM T93788 C6JZS7 62706349 EC50 = 270 nM T93788 C9QXO1 62706352 EC50 = 736 nM T93788 CN2XQ4 62706354 EC50 = 511 nM T93788 C13TEN 62706355 EC50 = 268 nM T93788 CLJ6A2 62706513 EC50 = 86 nM T93788 C2C4SU 62706514 EC50 = 770 nM T93788 C3P1WQ 62706516 EC50 = 550 nM T93788 CIB14P 62706517 EC50 = 1029 nM T93788 C53CKU 62706518 EC50 = 46 nM T93788 C8ALV4 62706691 EC50 = 272 nM T93788 CK6DX5 62706692 EC50 = 734 nM T93788 C9WVI6 62707006 EC50 = 58 nM T93788 CQ3R2L 66554587 EC50 = 505 nM T93788 C7KXP6 66554590 EC50 = 707 nM T93788 CJB58T 66554759 EC50 = 1030 nM T93788 CN62FS 66554760 EC50 = 38 nM T93788 C0S7TI 66554933 EC50 = 63 nM T93788 C80TYS 66556121 EC50 = 16 nM T93788 CL6E7G 66556122 EC50 = 57 nM T93788 C2TLX9 66556297 EC50 = 6.4 nM T93788 CKC76E 66556631 EC50 = 134 nM T93788 C4L7EO 66556985 EC50 = 42 nM T93788 C14BKV 66561292 EC50 = 33 nM T93788 CC6RH8 66574514 EC50 = 13.8 nM T93788 C7YQS4 66826123 EC50 = 100000000 nM T93788 CAS64Z 66963482 EC50 > 300 nM T93788 C0VD5C 66963512 EC50 = 20 nM T93788 CLB8H7 66963587 EC50 = 20 nM T93788 CFA02S 66963820 EC50 = 190 nM T93788 C41YUC 66963944 EC50 = 560 nM T93788 CBHA32 66963969 EC50 = 190 nM T93788 CCT84Y 66963996 EC50 = 4 nM T93788 CY8FU4 66964035 EC50 = 880 nM T93788 CM8X6G 66964040 EC50 = 3 nM T93788 CE10UM 66964044 EC50 = 170 nM T93788 CWA7I2 66964068 EC50 = 180 nM T93788 C6AU3Y 66964159 EC50 = 73 nM T93788 CI12ZB 66964172 EC50 = 243 nM T93788 CYB30V 66964174 EC50 = 1200 nM T93788 CXB50V 66964195 EC50 = 164 nM T93788 CB9U5D 66964295 EC50 = 10 nM T93788 CJQ0R1 66964459 EC50 = 86 nM T93788 CBP0V7 66964466 EC50 = 40 nM T93788 CE9DN2 66964510 EC50 = 11 nM T93788 CDO06R 66964555 EC50 = 1 nM T93788 CI4D3Q 66964595 EC50 > 10000 nM T93788 CM6QF7 66964599 EC50 = 40 nM T93788 CT2S3O 66964600 EC50 = 140 nM T93788 CH3KD5 66964621 EC50 = 290 nM T93788 CUI2X7 66964622 EC50 = 16 nM T93788 CR4O5S 66964658 EC50 = 340 nM T93788 CA6VM4 66964662 EC50 = 110 nM T93788 CG3WV5 66964682 EC50 = 1300 nM T93788 CWS5M3 66964756 EC50 = 130 nM T93788 CF35RW 66964802 EC50 = 62 nM T93788 CUA2J7 66964831 EC50 = 53 nM T93788 C1LY4J 66964852 EC50 = 63 nM T93788 CJ01UH 67449544 EC50 = 9.6 nM T93788 C73NJP 67449861 EC50 = 13 nM T93788 CGDH12 67449879 EC50 = 47 nM T93788 CQ4AN2 67450521 EC50 = 651 nM T93788 CO9M8S 67450901 EC50 = 427 nM T93788 C8OEN6 67450949 EC50 = 11 nM T93788 CFXC10 67451300 EC50 = 776 nM T93788 C20IRD 67606673 EC50 = 19.3 nM T93788 CG5E0I 67607375 EC50 = 15 nM T93788 CX45AB 67633261 EC50 = 2.78 nM T93788 CKHT83 67950429 EC50 = 5.32 nM T93788 CAT15Y 68021765 EC50 = 37 nM T93788 CHO94B 68021862 EC50 = 70 nM T93788 CXM35D 68021864 EC50 = 31 nM T93788 CUL1T2 68021959 EC50 = 21 nM T93788 C61YKH 68021978 EC50 = 52 nM T93788 CT1L6E 68022035 EC50 = 13 nM T93788 C7V0LF 68022196 EC50 = 63 nM T93788 C7AS8M 68022224 EC50 = 42 nM T93788 COG3A9 68022271 EC50 = 97 nM T93788 C95FCX 68036465 EC50 = 6 nM T93788 CI1DR8 68036798 EC50 = 49 nM T93788 C8L7PV 68036809 EC50 = 10 nM T93788 C2WJ4D 68036822 EC50 = 188 nM T93788 CZS1M5 68036918 EC50 = 26 nM T93788 C27XCG 68036931 EC50 = 10 nM T93788 CDM27X 68036951 EC50 = 19 nM T93788 CSE08J 68039954 EC50 = 4 nM T93788 C5WC9G 68040003 EC50 = 16 nM T93788 CCZ6Y5 68040038 EC50 = 7 nM T93788 CK21EZ 68040046 EC50 = 25 nM T93788 C0VHJ6 68211518 EC50 = 67 nM T93788 CVR1U4 68211526 EC50 = 82 nM T93788 C96SFV 68211777 EC50 = 5 nM T93788 COC2V7 68211779 EC50 = 78 nM T93788 CQ5X0V 68211781 EC50 = 122 nM T93788 COT43B 68211784 EC50 = 34 nM T93788 CIP2R1 68211791 EC50 = 2 nM T93788 C8SQA4 68211912 EC50 = 28 nM T93788 CY7NQ6 68211918 EC50 = 70 nM T93788 CF3VW9 68229751 EC50 = 52 nM T93788 CQPU67 68230018 EC50 = 36.8 nM T93788 CDPS39 68230201 EC50 = 8.3 nM T93788 CVA87O 68230212 EC50 = 3 nM T93788 CYV6B4 68230358 EC50 = 5.3 nM T93788 CA2YH5 68240224 EC50 = 70 nM T93788 C1TQ9C 68240419 EC50 = 7 nM T93788 CO8Z1E 68240486 EC50 = 51 nM T93788 CG3B4U 68299301 EC50 = 39 nM T93788 CU0A1F 68299305 EC50 = 240 nM T93788 CTQ78Y 68299308 EC50 = 1200 nM T93788 C14NSX 68385332 EC50 = 21 nM T93788 CN12IT 70680969 EC50 = 538 nM T93788 C0VEM7 70680970 EC50 = 441 nM T93788 CBE03K 70682125 EC50 = 254 nM T93788 C8D6ZB 70683088 EC50 > 30000 nM T93788 CKM4C2 70683089 EC50 = 1890 nM T93788 C7BPF4 70683090 EC50 = 29 nM T93788 CRTD40 70683091 EC50 = 29 nM T93788 CD0I2O 70684960 EC50 = 236 nM T93788 CKN95T 70685174 EC50 = 131 nM T93788 CUQ92A 70685175 EC50 = 172 nM T93788 CD7RB3 70687121 EC50 = 44 nM T93788 CY0N4S 70687331 EC50 = 122 nM T93788 C84GET 70687332 EC50 = 18 nM T93788 C6LN3I 70688972 EC50 = 78 nM T93788 CL68HK 70689385 EC50 = 1345 nM T93788 CBY8T6 70689386 EC50 = 53 nM T93788 CTJL92 70689387 EC50 = 485 nM T93788 CJY73E 70691486 EC50 = 456 nM T93788 CV8QT4 70691487 EC50 = 7 nM T93788 CJS34X 70692694 EC50 = 2610 nM T93788 CM4P5Z 70693582 EC50 = 489 nM T93788 CA9R2G 70693583 EC50 = 535 nM T93788 C35ASU 70693584 EC50 = 76 nM T93788 C8JUY5 70693585 EC50 = 396 nM T93788 CX0E3Y 70693586 EC50 = 12 nM T93788 C5T6JA 70695705 EC50 = 140 nM T93788 CG1XU6 70796891 EC50 = 17 nM T93788 C83TQO 70810684 EC50 = 200 nM T93788 CKP4O8 70855957 EC50 = 3.3 nM T93788 CLKU89 70856302 EC50 = 2 nM T93788 C2OH1E 71081343 EC50 = 142 nM T93788 CCXB25 71081352 EC50 = 56 nM T93788 C6DW7Q 71081378 EC50 > 1000 nM T93788 CTWH36 71081448 EC50 = 68 nM T93788 C2BND6 71081449 EC50 = 98 nM T93788 CY9IP1 71081450 EC50 = 46 nM T93788 CWC86N 71081517 EC50 = 369 nM T93788 C1XHA8 71116039 EC50 = 2.1 nM T93788 C4YJI5 71116044 EC50 = 1.1 nM T93788 C2M4CU 71116111 EC50 = 4.8 nM T93788 CWFL92 71116113 EC50 = 7.1 nM T93788 CI09HU 71128813 EC50 = 1.7 nM T93788 CDP0X1 71128816 EC50 = 3.1 nM T93788 CX15DJ 71134925 EC50 = 35 nM T93788 C4ZEN1 71135255 EC50 = 1.5 nM T93788 C6B2XM 71135993 EC50 = 47 nM T93788 C5AUY8 71136686 EC50 = 1.7 nM T93788 CY3N9S 71140721 EC50 = 2.5 nM T93788 CSEU81 71208589 EC50 = 2 nM T93788 CTQJ18 71208637 EC50 = 3 nM T93788 C2PSM5 71208866 EC50 = 3 nM T93788 CYK27V 71287378 EC50 = 386 nM T93788 CT51PO 71287404 EC50 = 103 nM T93788 C9OC0D 71450290 EC50 = 158.49 nM T93788 CZQE65 71452110 EC50 = 21 nM T93788 CRF56L 71453941 EC50 = 30 nM T93788 CLIA38 71455380 EC50 = 630.96 nM T93788 CF8EI7 71455832 EC50 = 2 nM T93788 C52GYP 71457626 EC50 = 228 nM T93788 C94UFY 71459020 EC50 > 10000 nM T93788 C1AS4O 71459320 EC50 = 93 nM T93788 CP32HG 71459321 EC50 = 398.11 nM T93788 CXZ79V 71461092 EC50 = 501.19 nM T93788 C7RH2E 71462834 EC50 = 800 nM T93788 C2AY8E 71462835 EC50 = 100 nM T93788 CKOZ97 71471638 EC50 = 82 nM T93788 CV78KN 71471711 EC50 = 3 nM T93788 CYT2N9 71471779 EC50 = 26 nM T93788 CAQ08G 71471851 EC50 = 781 nM T93788 C9JV4A 71474021 EC50 = 2.3 nM T93788 CW4UL3 71474456 EC50 = 8.7 nM T93788 CDO0M1 71491707 EC50 = 25 nM T93788 C3MK2J 71491755 EC50 = 67 nM T93788 CDR72Y 71519025 EC50 > 10000 nM T93788 C7CW1F 71519026 EC50 = 240 nM T93788 CJ29OT 71519027 EC50 = 462 nM T93788 C5LV7I 71519189 EC50 = 260 nM T93788 C9F2HA 71519190 EC50 = 864 nM T93788 CIRC04 71519192 EC50 = 83 nM T93788 C5L7YM 71519193 EC50 = 498 nM T93788 CZ0O9G 71524800 EC50 > 10000 nM T93788 C4E0UB 71524801 EC50 > 10000 nM T93788 C1GOB4 71524802 EC50 > 10000 nM T93788 CPC67E 71524845 EC50 > 10000 nM T93788 CX0HP2 71524846 EC50 > 10000 nM T93788 C62LOK 71524848 EC50 > 10000 nM T93788 CO2PS5 71524849 EC50 > 10000 nM T93788 CM2A0F 71531541 EC50 = 14 nM T93788 C34LHD 71545377 EC50 = 559 nM T93788 C3WM2U 71545378 Ki = 1970 nM T93788 C3KF1D 71545379 Ki = 586 nM T93788 C6HC8D 71545380 EC50 = 130 nM T93788 CGR96T 71545381 EC50 = 40 nM T93788 CK2R7U 71545535 EC50 = 88 nM T93788 CV15FW 71545536 EC50 = 145 nM T93788 C6JDU1 71545537 EC50 = 155 nM T93788 C09LAW 71545538 EC50 = 75 nM T93788 C3SB6R 71545698 EC50 = 40 nM T93788 CD9PH4 71545699 EC50 = 121 nM T93788 C87LNP 71545700 Ki = 131 nM T93788 CSP17W 71546032 Ki > 8148 nM T93788 C6C9MQ 71546033 Ki > 8148 nM T93788 C20IJM 71546034 EC50 = 164 nM T93788 CVQO13 71546035 EC50 = 49 nM T93788 CP9I5A 71546036 EC50 = 16 nM T93788 CMGZ54 71546198 Ki > 7318 nM T93788 CY7D8H 71546199 Ki = 814 nM T93788 C75OBG 71546200 EC50 = 691 nM T93788 CMX3O9 71546201 EC50 = 1028 nM T93788 C5GEA2 71546202 EC50 = 144 nM T93788 C5PS7U 71546701 EC50 = 274 nM T93788 C2GTU1 71546853 Ki = 133 nM T93788 C5E2DN 71546854 EC50 = 202 nM T93788 CVU95B 71546855 Ki = 94 nM T93788 C0K7MN 71546856 EC50 = 39 nM T93788 CUC38V 71546857 EC50 = 17 nM T93788 CZQ7I0 71547006 Ki = 18 nM T93788 CYG0K4 71547007 Ki = 15 nM T93788 CIL7K6 71547008 Ki = 7 nM T93788 CATD09 71547153 EC50 = 1049 nM T93788 CFO9U7 71562723 EC50 = 11.5 nM T93788 C4NYA9 71562724 EC50 = 1.5 nM T93788 C8SX0I 71562725 EC50 > 10000 nM T93788 CPDO92 71562726 EC50 = 6.7 nM T93788 C4IMF0 71562845 EC50 = 4.9 nM T93788 C0QF2W 71562846 EC50 = 1.4 nM T93788 CB2F3M 71573174 EC50 = 0.8 nM T93788 CFD8Y0 71617876 EC50 > 1000 nM T93788 CLV15A 71654936 EC50 = 8400 nM T93788 C7ZT6C 71654937 EC50 = 660 nM T93788 C73QOD 71654938 EC50 = 810 nM T93788 CSO8Q5 71654939 EC50 = 270 nM T93788 C6LB8Q 71654940 EC50 = 380 nM T93788 C0SL8O 71655012 EC50 = 960 nM T93788 C0CEI6 71655013 EC50 = 1600 nM T93788 CP5U6A 71655014 EC50 = 380 nM T93788 C1F7DV 71655015 EC50 = 440 nM T93788 C5U2SI 71655016 EC50 = 1710 nM T93788 CS5C9G 71655017 EC50 = 2120 nM T93788 CN1O2A 71655092 EC50 = 2060 nM T93788 C9F8JQ 71655093 EC50 = 13 nM T93788 CJ2C0H 71655094 EC50 = 130 nM T93788 CATY06 71655095 EC50 = 4000 nM T93788 CV3E0U 71655096 EC50 = 2740 nM T93788 C2KQM7 71655097 EC50 = 31 nM T93788 CRM32P 71655175 EC50 = 350 nM T93788 CNP0B9 71655176 EC50 = 2950 nM T93788 C3YWF0 71655177 EC50 = 610 nM T93788 C9FNO1 71655178 EC50 = 50 nM T93788 C40DNC 71655179 EC50 = 16 nM T93788 C7WPG4 71655180 EC50 = 160 nM T93788 CAKV27 71655250 EC50 = 450 nM T93788 C31RYO 71655251 EC50 = 91 nM T93788 C6MP4D 71655252 EC50 = 68 nM T93788 C73IXR 71655253 EC50 = 89 nM T93788 C38LKC 71655254 EC50 = 300 nM T93788 CUB71C 71655255 EC50 = 1060 nM T93788 C4LP8D 71655315 EC50 = 20 nM T93788 CC2E1S 71713968 EC50 = 45 nM T93788 CD19YH 71716097 Ki = 33 nM T93788 CV17DK 71716738 EC50 = 47 nM T93788 C8O5AK 71717057 EC50 > 10000 nM T93788 CO2B1U 71717058 EC50 > 10000 nM T93788 CC3L9V 71717059 EC50 = 1000 nM T93788 CM68ZB 71717312 Ki = 125 nM T93788 CUV09L 71717324 EC50 = 300 nM T93788 C57MSH 71717334 EC50 = 181 nM T93788 CHDN36 71717681 EC50 > 10000 nM T93788 CT02GM 71718289 EC50 = 1000 nM T93788 CH8J2D 71718290 EC50 > 10000 nM T93788 CGBW84 71718892 EC50 > 10000 nM T93788 CL28YO 71719746 Ki = 948 nM T93788 CZ7BL8 71720095 EC50 > 10000 nM T93788 CW4M7K 71720096 EC50 = 1000 nM T93788 CPMS07 71720493 EC50 = 38 nM T93788 C9F0ZD 71720494 EC50 = 15 nM T93788 C4OL0Q 71720750 EC50 > 10000 nM T93788 C68DRE 71720751 EC50 > 10000 nM T93788 C30NBJ 71722055 EC50 = 11 nM T93788 CP2EY7 72188621 EC50 = 20 nM T93788 CF9I2U 72945517 EC50 = 19 nM T93788 CZQL46 72945518 EC50 = 15 nM T93788 CH1DA7 72945519 EC50 = 121 nM T93788 CM7EQ0 72945706 EC50 = 23 nM T93788 CH3KN2 72945707 EC50 = 11 nM T93788 C4B3SM 72945708 EC50 = 13 nM T93788 CYE12L 72945709 EC50 = 69 nM T93788 C23YTU 72945710 EC50 = 299 nM T93788 CG28EU 72945711 EC50 = 19 nM T93788 CGV82Z 72945895 EC50 = 224 nM T93788 C64CUT 72945896 EC50 = 382 nM T93788 CT93UL 72945897 EC50 = 238 nM T93788 CF39JH 72945898 EC50 > 30000 nM T93788 CNEP39 72945899 EC50 = 11 nM T93788 CQD6X0 72945900 EC50 = 9 nM T93788 CK5F2R 72946091 EC50 = 33 nM T93788 COEL45 72946092 EC50 = 16 nM T93788 CQ0I8V 72946093 EC50 = 357 nM T93788 CZMF40 72946094 EC50 = 493 nM T93788 CGK87R 73348101 EC50 = 630.96 nM T93788 CNM19T 73348866 EC50 = 7 nM T93788 CEF4B6 73350444 IC50 = 1 nM T93788 C5ON3C 73351961 EC50 = 11 nM T93788 CA95TW 73353419 EC50 = 6 nM T93788 CG7R3F 73353420 IC50 = 8 nM T93788 CB9YC7 73354930 EC50 = 79 nM T93788 CS90NU 73354931 IC50 = 3 nM T93788 C46PFQ 73357217 EC50 = 50.12 nM T93788 CK9T1Y 76309728 EC50 = 18 nM T93788 C2FUH7 76309729 EC50 = 131 nM T93788 CJ2M6A 76309730 EC50 = 61 nM T93788 CHK8N4 76309731 EC50 = 37 nM T93788 C8GA1B 76309732 EC50 = 32 nM T93788 C7FA4M 76309733 EC50 = 44 nM T93788 CP98VM 76310374 EC50 = 190 nM T93788 CRF25S 76310375 EC50 = 80 nM T93788 CIC5H2 76310376 EC50 = 100 nM T93788 CLW2K8 76310377 EC50 = 590 nM T93788 CP2C1O 76310397 EC50 = 120 nM T93788 CG35AY 76310438 EC50 = 2600 nM T93788 CZMC38 76310439 EC50 = 8.4 nM T93788 CEUA45 76310440 EC50 = 25 nM T93788 CPN8X0 76310441 EC50 = 21 nM T93788 C9FHP1 76310464 EC50 = 520 nM T93788 CLM1B6 76313416 EC50 = 15 nM T93788 CBQN52 76314040 EC50 = 70 nM T93788 CBA5Y4 76314041 EC50 = 310 nM T93788 C2RBC6 76314042 EC50 = 30 nM T93788 C0BO3U 76314043 EC50 = 100 nM T93788 CSR01W 76314044 EC50 = 50 nM T93788 C71KTD 76314045 EC50 = 290 nM T93788 CC0T9X 76314046 EC50 = 550 nM T93788 CQZ42U 76314047 EC50 = 540 nM T93788 CEX20O 76314048 EC50 = 90 nM T93788 C5GX3R 76314049 EC50 = 100 nM T93788 C1Y7ST 76314096 EC50 = 770 nM T93788 C3WX7M 76314115 EC50 = 3.9 nM T93788 C6O9DC 76316923 EC50 = 30 nM T93788 CWY57O 76316924 EC50 = 30 nM T93788 CEKG37 76316925 EC50 = 330 nM T93788 CF2P0G 76316926 EC50 > 5000 nM T93788 CH4C1Q 76316927 EC50 = 112 nM T93788 CL1CQ3 76316928 EC50 = 2120 nM T93788 C7RMQ3 76316929 EC50 > 30000 nM T93788 C8HM5Q 76317599 EC50 = 140 nM T93788 CZE2C1 76317600 EC50 = 40 nM T93788 C6RSN9 76317666 EC50 = 4800 nM T93788 CMYI68 76317689 EC50 = 44 nM T93788 CF9YM4 76317690 EC50 = 490 nM T93788 CZAG95 76320654 EC50 = 24 nM T93788 C70EDY 76320655 EC50 = 15 nM T93788 CFP85B 76320656 EC50 = 166 nM T93788 CFH1N6 76320657 EC50 = 50 nM T93788 C92DQF 76320658 EC50 = 34 nM T93788 CG28EB 76320659 EC50 = 18 nM T93788 CSAO79 76321321 EC50 = 80 nM T93788 C1GY3S 76321322 EC50 = 50 nM T93788 C8JI2C 76321323 EC50 = 80 nM T93788 CH01KT 76321324 EC50 = 4300 nM T93788 CF3JM5 76321325 EC50 = 180 nM T93788 CX7LQ3 76321373 EC50 = 2400 nM T93788 CZM0K5 76324299 EC50 = 112 nM T93788 CN60XY 76324300 EC50 = 42 nM T93788 C9AG5H 76324301 EC50 = 54 nM T93788 CS6MC7 76324302 EC50 = 38 nM T93788 C0QNR4 76324928 EC50 = 110 nM T93788 CH8MK5 76324929 EC50 = 80 nM T93788 CWAX90 76324930 EC50 = 1500 nM T93788 C3JZU2 76324931 EC50 = 50 nM T93788 C6C5OD 76324932 EC50 = 270 nM T93788 CD0P3F 76324933 EC50 = 90 nM T93788 CA3O5D 76324934 EC50 = 70 nM T93788 C0K9BQ 76324949 EC50 > 30000 nM T93788 CAH91F 76324976 EC50 = 120 nM T93788 C3P5HT 76324977 EC50 = 25 nM T93788 C43DST 76324996 EC50 = 1700 nM T93788 C26MHI 76327867 EC50 = 24 nM T93788 CP3VI7 76327868 EC50 = 38 nM T93788 CRC1N8 76328493 EC50 = 180 nM T93788 CBM47D 76328494 EC50 = 60 nM T93788 CQC2W3 76328495 EC50 = 60 nM T93788 CA7T2L 76328496 EC50 = 30 nM T93788 CM83BG 76328497 EC50 = 80 nM T93788 CLT09R 76328549 EC50 = 530 nM T93788 CN82FC 76328564 EC50 = 6.8 nM T93788 CA8JB0 76331519 EC50 = 25 nM T93788 CM4QH5 76331520 EC50 = 7 nM T93788 CT0RW4 76331521 EC50 = 86 nM T93788 CQFZ48 76332169 EC50 = 130 nM T93788 C8BZ5R 76332170 EC50 = 100 nM T93788 CV76UF 76332171 EC50 = 320 nM T93788 C40DUR 76332172 EC50 = 90 nM T93788 CWBF71 76332173 EC50 = 770 nM T93788 CH23MG 76332174 EC50 = 860 nM T93788 C0H6SK 76332225 EC50 = 68 nM T93788 C0XJO8 76335131 EC50 = 18 nM T93788 CF6S7P 76335814 EC50 = 100 nM T93788 C3BNF9 76335815 EC50 = 60 nM T93788 C28FTZ 76335830 EC50 = 270 nM T93788 CRZ07L 76335866 EC50 = 1400 nM T93788 CLE6X0 76335867 EC50 = 2500 nM T93788 CT4XY9 76335868 EC50 = 160 nM T93788 C1KL8Q 76683707 EC50 = 55 nM T93788 CA6XJ7 76683708 EC50 = 14 nM T93788 C9Z1TP 76683709 EC50 = 9 nM T93788 CQX8U3 76683715 EC50 = 31 nM T93788 CQH2D6 76683814 EC50 = 78 nM T93788 C0EK4U 76683914 EC50 = 48 nM T93788 C1EBJ5 76683917 EC50 = 8 nM T93788 CDGL78 76684031 EC50 = 52 nM T93788 C10CNR 76684033 EC50 = 29 nM T93788 CWQF87 76684133 EC50 = 63 nM T93788 CL9JB3 86566993 EC50 = 716 nM T93788 CLO4Z6 86709924 EC50 = 7.91 nM T93788 CUW93G 86717800 EC50 = 4.5 nM T93788 C2FP3R 87217189 EC50 = 58 nM T93788 CER7N3 88567661 EC50 = 17 nM T93788 C83JRE 89583782 EC50 = 1.8 nM T93788 C1ZPE2 89583933 EC50 = 9.4 nM T93788 CU74LB 89584002 EC50 = 0.2 nM T93788 CBQ8J0 89584012 EC50 = 0.8 nM T93788 CR0P6K 89584034 EC50 = 0.2 nM T93788 C4NZW1 89584050 EC50 = 1.5 nM T93788 CZOJ21 89584118 EC50 = 0.7 nM T93788 CG29VI 90115611 EC50 = 4.2 nM T93788 C75OYT 90116115 EC50 = 3.2 nM T93788 C0A7DJ 90148901 EC50 = 4.5 nM T93788 CPE2L1 90656488 EC50 = 9000 nM T93788 C7CPS9 90656489 EC50 = 1100 nM T93788 CO03AL 90656490 EC50 > 10000 nM T93788 CC48DN 90656491 EC50 > 10000 nM T93788 CYF04H 90656492 EC50 > 10000 nM T93788 C2I8LO 90656529 EC50 = 541 nM T93788 C1X2PV 90665949 EC50 = 25.12 nM T93788 CKY18S 90665950 EC50 = 158.49 nM T93788 C31ZSK 90666908 EC50 = 100 nM T93788 CXKO79 90666909 EC50 = 630.96 nM T93788 C1JB5U 90666910 EC50 = 15.85 nM T93788 C9W6EJ 90666911 EC50 = 199.53 nM T93788 CE5J4N 90666912 EC50 = 199.53 nM T93788 CI02ZU 90666913 EC50 = 199.53 nM T93788 CTP5L0 90666914 EC50 = 501.19 nM T93788 C5DJT8 90666915 EC50 = 1258.93 nM T93788 CL54KY 90666916 EC50 = 1584.89 nM T93788 C80DYO 91824767 EC50 = 5 nM T93788 C21PRZ 102361261 EC50 = 54 nM T93788 C8ZM9J 117678530 EC50 = 0.4 nM T93788 C5CL8X 117684497 EC50 = 2.2 nM T93788 C2QPR5 118709765 EC50 = 173 nM T93788 CGQ8K4 118709767 EC50 = 1200 nM T93788 CXG4W7 118709768 EC50 = 140 nM T93788 CT5Y4F 118711210 EC50 = 132 nM T93788 CFND64 118711211 EC50 = 21 nM T93788 C1K7AS 118711212 EC50 = 13.6 nM T93788 C9VIB0 118711213 EC50 = 6.53 nM T93788 CHJQ06 118711214 EC50 = 92.9 nM T93788 CD9CK6 118711215 EC50 = 19.9 nM T93788 CRZY56 118711216 EC50 = 65.5 nM T93788 CON5I0 118711217 EC50 = 196 nM T93788 C29OWT 118711218 EC50 = 186 nM T93788 CVK7D2 118711219 EC50 = 9.2 nM T93788 C9U2WG 118711775 EC50 = 9.86 nM T93788 COP9C4 118711776 EC50 = 22 nM T93788 C0J2QH 118711777 EC50 = 326 nM T93788 CA21CR 118711778 EC50 = 14.3 nM T93788 CQS5M1 118711779 EC50 = 29.3 nM T93788 CTL50A 118711780 EC50 = 6.8 nM T93788 C65LOQ 118711781 EC50 = 4.83 nM T93788 CSL1I4 118711782 EC50 = 24.9 nM T93788 C09AEX 118711783 EC50 = 13.2 nM T93788 C27LYA 118711784 EC50 = 8.51 nM T93788 CDJ1I4 118711785 EC50 = 69.9 nM T93788 C8R6MZ 118711787 EC50 = 151 nM T93788 C2EH6Z 118711788 EC50 = 37 nM T93788 C65TWF 118711789 EC50 = 76.3 nM T93788 C02WJT 118711790 EC50 = 17.4 nM T93788 CHC73U 118711791 EC50 = 24.7 nM T93788 C7IF1L 118711792 EC50 = 72.8 nM T93788 CB67JI 118711793 EC50 = 761 nM T93788 C2QRV5 118711794 EC50 = 21.2 nM T93788 CM4R6H 118711795 EC50 = 14 nM T93788 CDO2R1 118711796 EC50 = 43.4 nM T93788 C9OZK0 118711797 EC50 = 4.7 nM T93788 C0RM8O 118711798 EC50 = 6.12 nM T93788 CJ3U7V 118715130 EC50 > 10000 nM T93788 CFES75 118715131 EC50 > 10000 nM T93788 C46OKY 118715132 EC50 > 10000 nM T93788 CG6C2I 118715133 EC50 > 10000 nM T93788 C9IPD5 118715134 EC50 > 10000 nM T93788 CV7I4Q 118715135 EC50 > 10000 nM T93788 CS6CW7 118720403 EC50 > 10 nM T93788 CQ6ND5 118720404 EC50 = 23 nM T93788 C96JBI 118720405 EC50 = 0.5 nM T93788 CJQ58U 118720406 EC50 = 38 nM T93788 C4Y0OG 118720407 EC50 = 2 nM T93788 CF7NW4 118720408 EC50 = 3 nM T93788 C6BP7I 118720409 EC50 = 8 nM T93788 CBT12E 118720410 EC50 = 74 nM T93788 CYC0Q6 118720411 EC50 = 101 nM T93788 C08BWN 118720412 EC50 = 3 nM T93788 CP95WQ 118720413 EC50 = 125 nM T93788 CEZK35 118720414 EC50 = 7 nM T93788 CP9JI8 118720415 EC50 = 20 nM T93788 CUNM53 118720416 EC50 = 11 nM T93788 CKX32F 118720417 EC50 = 25 nM T93788 CMX50B 118720418 EC50 = 34 nM T93788 C9BEO3 118720419 EC50 = 3 nM T93788 C0N4CQ 118720420 EC50 = 214 nM T93788 CM8F5R 118720421 EC50 = 73 nM T93788 CP2C9I 118720422 EC50 = 298 nM T93788 CG0VK4 118720423 EC50 = 2 nM T93788 C5CI4Z 118720424 EC50 = 436 nM T93788 CW50AC 118720425 EC50 = 21 nM T93788 C57HWX 118720426 EC50 = 15 nM T93788 C8XDH9 118720427 EC50 = 530 nM T93788 COB3W5 118720428 EC50 = 2 nM T93788 CVXN53 118720429 EC50 = 35 nM T93788 CP4SV0 118720430 EC50 = 20 nM T93788 CF87IO 118720431 EC50 = 2 nM T93788 CY6HT5 118720432 EC50 = 6 nM T93788 CPC71H 118722570 EC50 = 21 nM T93788 CTL19H 118722571 EC50 = 55 nM T93788 C2JGB3 118722572 EC50 = 10 nM T93788 CKD42B 118722573 EC50 = 133 nM T93788 C6PMQ1 118722574 EC50 = 150 nM T93788 C3ZL5Y 118722575 EC50 = 15 nM T93788 CR3UB2 118722576 EC50 = 7 nM T93788 CX1W8N 118722577 EC50 = 27 nM T93788 C49DXR 118722578 EC50 = 4 nM T93788 CW5GK1 118722579 EC50 = 58 nM T93788 C50GXM 118722580 EC50 = 158 nM T93788 CEI62G 118722581 EC50 = 4 nM T93788 C9UG3Z 118722582 EC50 = 8 nM T93788 C5XH4V 118722583 EC50 = 91 nM T93788 C6Q3RV 118722584 EC50 = 1102 nM T93788 CCWD82 118722585 EC50 = 4 nM T93788 CZ0DG2 118722586 EC50 = 18 nM T93788 CI3R9V 118722587 EC50 = 6 nM T93788 C6Z4FK 122184143 EC50 = 38.4 nM T93788 CP80EY 122184144 EC50 = 107 nM T93788 C4MZF8 122184145 EC50 = 48.8 nM T93788 CR9O1L 122184146 EC50 = 291 nM T93788 CZS80P 122184147 EC50 = 14 nM T93788 CHY08E 122184148 EC50 = 9.1 nM T93788 C07AXY 122184149 EC50 = 10.7 nM T93788 CQT12A 122184150 EC50 = 30.3 nM T93788 CP42FU 122184151 EC50 > 100000 nM T93788 CIB30N 122191630 EC50 = 3.3 nM T93788 CYI12O 122191631 EC50 = 2.4 nM T93788 CW1NI3 122191632 EC50 = 1.7 nM T93788 C5GRC3 122191633 EC50 = 0.8 nM T93788 CCTM93 122194337 EC50 = 17 nM T93788 C9MBL0 122194338 EC50 = 44 nM T93788 C7C4WK 122194339 EC50 = 65 nM T93788 CXAK04 122194420 EC50 = 5 nM T93788 CXV30P 122194421 EC50 = 268 nM T93788 C0DFN8 127048479 EC50 = 177 nM T93788 CIC9S6 127048480 EC50 = 266 nM T93788 CQL9H0 127048481 EC50 = 197 nM T93788 CRY0I8 127048482 EC50 = 27 nM T93788 CW09RY 127048491 EC50 = 46 nM T93788 C97SDN 127048492 EC50 = 10 nM T93788 CHT2M6 127048493 EC50 = 14 nM T93788 CQIB34 127048494 EC50 = 92 nM T93788 C2V1CS 127048495 EC50 = 11 nM T93788 CP7Y0X 127048787 EC50 = 20 nM T93788 C0XV9A 127048820 EC50 = 23 nM T93788 CP6C2G 127048821 EC50 = 30 nM T93788 CX7K0M 127048822 EC50 = 220 nM T93788 CK1R4X 127050518 EC50 = 10 nM T93788 C0EN7J 127050519 EC50 = 4 nM T93788 C04MCY 127050520 EC50 = 15 nM T93788 C5DA9S 132486941 EC50 = 65 nM T93788 CY4FW5 134131905 EC50 = 1.3 nM T93788 CMY0V5 134132485 EC50 = 1900 nM T93788 C1T4DP 134134925 EC50 > 2000 nM T93788 C6R3US 134135618 EC50 = 1.6 nM T93788 CVE5Z8 134136399 EC50 = 0.6 nM T93788 CTZ0Y6 134136992 EC50 = 44.2 nM T93788 CRL94F 134137238 EC50 > 2000 nM T93788 C6UXF4 134138752 EC50 = 6.2 nM T93788 CY2HZ6 134139363 EC50 > 2000 nM T93788 C1JF9T 134139552 EC50 > 2000 nM T93788 CY9RM8 134142930 EC50 = 1.5 nM T93788 CFG3B4 134146906 EC50 > 2000 nM T93788 C9KWZ2 134147816 EC50 = 3.5 nM T93788 CZSA25 134147992 EC50 = 1.5 nM T93788 C8ALS5 134150100 EC50 > 2000 nM T93788 C0G5PV 134151859 EC50 = 950 nM T93788 C5U4GE 134152907 EC50 = 205 nM T93788 C4XS1N 134156472 EC50 > 2000 nM T93788 C3MU5V 134156958 EC50 = 1.4 nM T93788 CIRH31 137631474 EC50 = 61 nM T93788 CF8W4G 137631845 EC50 = 4.9 nM T93788 CCM7B3 137632132 EC50 = 5.6 nM T93788 C2B8YF 137632493 EC50 = 98 nM T93788 CINX05 137632674 EC50 = 48.2 nM T93788 C8J9AS 137632950 EC50 = 9 nM T93788 CF9QR4 137632997 EC50 = 171 nM T93788 CW9R5V 137633747 EC50 = 10 nM T93788 C3BCO0 137633771 EC50 = 252 nM T93788 C6PU4J 137634756 EC50 = 793 nM T93788 CV5E4H 137634873 EC50 = 3.1 nM T93788 CT72HP 137635337 EC50 = 310 nM T93788 CY10HA 137637825 EC50 = 5.6 nM T93788 C50UHW 137637873 EC50 = 27 nM T93788 CNI5D0 137637925 EC50 = 199 nM T93788 C9P7HM 137637929 EC50 = 18 nM T93788 CJX6U4 137638009 EC50 = 155 nM T93788 C78HPO 137638017 EC50 = 73 nM T93788 CGA3P4 137638546 EC50 > 10000 nM T93788 CWYG89 137639896 EC50 = 60 nM T93788 CM3VF9 137639995 EC50 = 92 nM T93788 CEYK56 137641046 EC50 = 39 nM T93788 C7K9VU 137642901 EC50 = 586 nM T93788 CYOZ07 137642936 EC50 = 64 nM T93788 CHA47F 137643188 EC50 = 19 nM T93788 CQ5DI1 137643239 EC50 = 67 nM T93788 C7AJG1 137643726 EC50 = 77 nM T93788 C7SH2E 137643838 EC50 = 315 nM T93788 C4EMC3 137643882 EC50 = 321 nM T93788 CH1P4Y 137643950 EC50 > 1000 nM T93788 CUGP54 137645678 EC50 = 391 nM T93788 CV4H9N 137645720 EC50 = 110 nM T93788 CB8CX4 137647821 EC50 = 82 nM T93788 CY7OR0 137648824 EC50 = 105 nM T93788 CEYZ80 137648888 EC50 = 201 nM T93788 C7BXJ2 137649810 EC50 = 1.8 nM T93788 CJVM79 137650572 EC50 = 53 nM T93788 C4F9GB 137651939 EC50 = 83 nM T93788 CHQI31 137651954 EC50 = 512 nM T93788 C3QD8P 137651958 EC50 = 2 nM T93788 C0E5FI 137653591 EC50 = 77.7 nM T93788 CPR76C 137655251 EC50 = 7 nM T93788 C97RZV 137655380 EC50 = 319 nM T93788 C1W9SE 137656527 EC50 = 53 nM T93788 CU9KZ4 137656911 EC50 = 15 nM T93788 CMF10H 137656947 EC50 = 78 nM T93788 CL9VW3 137657254 EC50 = 156 nM T93788 CNE31G 137659062 EC50 = 18 nM T93788 CS6G8H 137659500 EC50 = 1.2 nM T93788 CTK8D1 137660158 EC50 = 67 nM T93788 CI7Q4L 137660484 EC50 = 57 nM T93788 C1BXZ4 137660724 EC50 = 83 nM T93788 C7L5MD 137661403 EC50 = 13 nM T93788 C30NUT 137661559 EC50 = 33 nM T93788 CW1VR8 139436992 EC50 = 12 nM T93788 C9MX3E 139437014 EC50 = 4920 nM T93788 CB5Q2E 139437017 EC50 = 57 nM T93788 CO7T8R 139437037 EC50 = 458 nM T93788 CLO92I 139437040 EC50 = 82 nM T93788 C6BW7F 139437096 EC50 = 324 nM T93788 C0KI5D 140251500 EC50 = 31 nM T93788 CAE54O 140251501 EC50 = 13 nM T93788 CQA4W0 140251511 EC50 = 23 nM T93788 C2K4QW 140251527 EC50 = 40 nM T93788 CA5CF8 140251528 EC50 = 18 nM T93788 CU2ND3 140251533 EC50 = 34 nM T93788 C2VA1I 140253894 EC50 = 101 nM T93788 C8Z2XA 140253895 EC50 = 128 nM T93788 CT6D1A 140253898 EC50 = 17 nM T93788 CNQ53I 140254089 EC50 = 235 nM T93788 C8T6NF 140254101 EC50 = 169 nM T93788 CING28 144479903 EC50 = 334 nM T93788 C2OX1H 145949313 EC50 = 5.1 nM T93788 C0M3YQ 145949889 EC50 = 97 nM T93788 CYOH06 145951687 EC50 = 212 nM T93788 CQX3I6 145955539 EC50 = 13 nM T93788 CWIC73 145957126 EC50 = 10 nM T93788 CKW4D7 145959739 EC50 = 3.5 nM T93788 CJD7L6 145962089 EC50 = 6 nM T93788 CJF21C 145963524 EC50 = 8 nM T93788 CPL94Z 145964295 EC50 = 21 nM T93788 C1YM2B 145964891 EC50 = 82 nM T93788 C85JQK 145964999 EC50 = 211 nM T93788 CH6R3O 145965514 EC50 = 182 nM T93788 C4ZM3X 145966434 EC50 = 100 nM T93788 C6SX5I 145966749 EC50 = 7 nM T93788 CZ1IP0 145967361 EC50 = 18 nM T93788 C4ZTN9 145967591 EC50 = 225 nM T93788 CT0WU8 145967680 EC50 = 830 nM T93788 CZKG72 145968038 EC50 = 1.995 nM T93788 CTI20V 145968103 EC50 = 2388 nM T93788 CF61IA 145968330 EC50 = 123 nM T93788 C7UK3H 145968709 EC50 = 49 nM T93788 CJ0KF3 145968993 EC50 = 2590 nM T93788 CIB03W 145969583 EC50 = 154 nM T93788 CSUM19 145969910 EC50 = 5.012 nM T93788 CB23AP 145970094 EC50 = 511 nM T93788 CFO6S8 145970276 EC50 = 19 nM T93788 CC5I3B 145970536 EC50 = 157 nM T93788 CU3PZ7 145970589 EC50 = 348 nM T93788 C8VGL2 145971166 EC50 = 183 nM T93788 C5HW3K 145971825 EC50 = 88 nM T93788 C1RCP7 145972319 EC50 = 10 nM T93788 CA31ZR 145973091 EC50 = 14 nM T93788 CCT96L 145973632 EC50 = 2.6 nM T93788 C0VY7G 145974170 EC50 = 95 nM T93788 C3KXP2 145975486 EC50 = 5 nM T93788 CPD46L 145975897 EC50 = 240 nM T93788 CQ2H6F 145976125 EC50 = 4 nM T93788 CS15QM 145976269 EC50 = 29 nM T93788 C3A5RU 145976366 EC50 = 27 nM T93788 CR42QN 145977018 EC50 = 4 nM T93788 C1CF9N 145978481 EC50 = 209 nM T93788 CFXA96 145978767 EC50 = 78 nM T93788 CV21OC 145978800 EC50 = 780 nM T93788 C8WE1P 145982637 EC50 = 8.1 nM T93788 C3ILT5 145983137 EC50 = 36 nM T93788 CPS7J2 145983474 EC50 = 44 nM T93788 CAR8P2 145983613 EC50 = 1000 nM T93788 CV06WH 145983959 EC50 > 10000 nM T93788 CS3V1K 145983970 EC50 = 3200 nM T93788 C2FZP3 145984093 EC50 = 2.2 nM T93788 CT8R0W 145984643 EC50 = 126 nM T93788 CHX51B 145985013 EC50 = 179 nM T93788 CN9B7H 145985036 EC50 = 2100 nM T93788 CQW14Z 145985107 EC50 = 345 nM T93788 CG97IV 145986139 EC50 = 49 nM T93788 C4L2EY 145986191 EC50 = 147 nM T93788 C7J6XS 145986357 EC50 = 25.12 nM T93788 C7GK3H 145990715 EC50 > 100000 nM T93788 CEA10I 145993111 EC50 = 321 nM T93788 CA8HW6 145993236 EC50 = 360 nM T93788 CM25YZ 155511104 EC50 = 4.21 nM T93788 C4HCA5 155513850 EC50 = 3.12 nM T93788 CV68IT 155514874 EC50 = 64 nM T93788 CCT2U1 155514929 EC50 = 29 nM T93788 CCA49B 155515010 EC50 = 44 nM T93788 C1XLC0 155515632 EC50 = 98 nM T93788 CVM52W 155516183 EC50 = 2457 nM T93788 CIT8G6 155517437 EC50 = 139 nM T93788 CM2F9X 155517636 EC50 = 8.78 nM T93788 C2XQY5 155521067 EC50 = 7 nM T93788 CK02AF 155522754 EC50 = 85 nM T93788 CCP59K 155523981 EC50 = 13.98 nM T93788 C03QFB 155524213 EC50 = 86 nM T93788 C24HCO 155525761 EC50 = 12.34 nM T93788 C5E1PD 155525764 EC50 = 31 nM T93788 CIP62K 155525822 EC50 = 7.12 nM T93788 C62FVA 155527157 EC50 = 25 nM T93788 CGP1Y7 155528031 EC50 = 15 nM T93788 C5OQV0 155528272 EC50 = 12.31 nM T93788 CQA30H 155528891 EC50 = 12.43 nM T93788 CDOI91 155530128 EC50 = 59 nM T93788 C70MHT 155530371 EC50 = 13.56 nM T93788 C2FO7T 155531204 EC50 = 261 nM T93788 CQ1OH3 155531494 EC50 = 5 nM T93788 CPH54I 155532104 EC50 = 301 nM T93788 CQ1F0P 155532657 EC50 = 89 nM T93788 CH6XR0 155532730 EC50 = 42 nM T93788 CYKT59 155534233 EC50 = 13 nM T93788 CU48LF 155536150 EC50 = 11.12 nM T93788 CCH57L 155537620 EC50 = 3.67 nM T93788 CYP63K 155537900 EC50 > 1000 nM T93788 C3PWV4 155538381 EC50 = 69 nM T93788 CEVC80 155538763 EC50 = 27 nM T93788 CF72OA 155539620 EC50 = 27 nM T93788 C7IMF1 155541499 EC50 > 1000 nM T93788 CS40NT 155542312 EC50 = 8.17 nM T93788 CGP4Z6 155544367 IC50 = 4620 nM T93788 CH25ZD 155549064 EC50 = 6 nM T93788 C16QAN 155550456 EC50 = 720 nM T93788 CQ14SC 155551991 EC50 = 33 nM T93788 CWP6G5 155553659 EC50 = 16 nM T93788 C2CD7U 155564944 EC50 = 426 nM T93788 CX7G8Q 155565475 EC50 = 3.59 nM T93788 CRV9Y2 155566096 EC50 = 430 nM T93788 CSK6A1 155566114 EC50 = 5 nM T93788 CAP48C 155567012 EC50 = 45 nM T93788 CX4O7N 155568284 EC50 = 10.43 nM T93788 CMC2A9 155568311 EC50 = 19 nM T93788 CSZ7N9 155569398 EC50 = 39 nM T93788 D00GTC 5332859 EC50 = 2500 nM T93788 D01GPC 53235534 EC50 = 4 nM T93788 D01VZL 11462546 EC50 = 1900 nM T93788 D06QYM 51346816 EC50 = 80 nM T93788 D07MBC 5283454 EC50 = 2200 nM T93788 D08HOK 11282871 EC50 = 1.1 nM T93788 D09ROS 54582152 EC50 = 0.6 nM T93788 D0I2EL 53630394 EC50 = 0.9 nM T93788 D0R5QF 24939268 EC50 = 0.65 nM T93788 D0VA7C 54580880 EC50 = 3600 nM T93788 D0X3NW 53630410 EC50 = 0.5 nM T50688 D07XHO 4413 IC50 = 12000 nM T50688 D09ZIO 448812 IC50 = 570 nM T50688 D0BN9X 60947 IC50 = 0.37 nM T50688 D0GY5Z 2244 IC50 = 5000 nM T50688 D01TJY 53340771 IC50 > 10 nM T50688 D09ZXO 176873 IC50 = 590 nM T50688 D0Q5LF 9961766 IC50 > 100000 nM T50688 D00VAJ 178080 IC50 = 2.38 nM T50688 D01QQM 3038484 IC50 = 1.4 nM T50688 D02VIP 9955461 Ki = 3300 nM T50688 D03GCN 9885190 IC50 = 25 nM T50688 D03QHI 9933077 IC50 = 0.4 nM T50688 D05JXR 9805266 IC50 = 72 nM T50688 D06LGC 9906649 IC50 = 50 nM T50688 D07EXV 60957 IC50 = 2 nM T50688 D08CQL 164393 Ki = 2 nM T50688 D08LIG 153986 IC50 > 3 nM T50688 D0B9SR 9868426 Ki = 3800 nM T50688 D0C7JH 6918252 IC50 = 29 nM T50688 D0D7GE 9824171 IC50 = 0.49 nM T50688 D0H1PN 9955286 IC50 = 4.7 nM T50688 D0I7EU 9827266 Ki = 1.6 nM T50688 D0K0NP 9812185 IC50 = 12 nM T50688 D0LK9N 66000 IC50 = 80 nM T50688 D0LT1S 9823503 Ki = 30000 nM T50688 D0M6YE 44343680 Ki = 175 nM T50688 D0N0BI 5491394 IC50 = 1.14 nM T50688 D0P8JX 177831 IC50 = 32 nM T50688 D0S3RB 216230 IC50 = 0.06 nM T50688 D0SV7D 80274 IC50 = 28 nM T50688 D0U4ZY 10031011 IC50 = 6 nM T50688 D0U6BB 44343739 IC50 = 94 nM T50688 D0W4OL 132814 IC50 = 88 nM T50688 D0Y0AP 173614 IC50 = 7.943 nM T50688 D0Z0XQ 44343754 IC50 = 30 nM T50688 D0Z9LD 9804438 IC50 = 1600 nM T50688 C7CL3Y 107775 IC50 = 7900 nM T50688 CE19HD 132605 IC50 = 1700 nM T50688 C0XC5J 164450 IC50 = 120 nM T50688 C81ZQR 164519 IC50 = 30 nM T50688 CFQU71 177231 IC50 = 0.25 nM T50688 C5HE6N 446808 IC50 = 12500 nM T50688 CE5LI6 448813 IC50 = 19 nM T50688 C7M9QB 756604 IC50 = 9600 nM T50688 C2E9ZX 3080994 IC50 = 31 nM T50688 CJ2PE8 3081210 Ki = 4200 nM T50688 CY7WS4 9799158 IC50 = 1000 nM T50688 CU7VY5 9800226 IC50 = 8500 nM T50688 C2ST5A 9801767 IC50 = 6 nM T50688 CS40VO 9802158 IC50 = 5500 nM T50688 C86OSU 9802663 IC50 > 10000 nM T50688 CH19JX 9804758 IC50 > 10000 nM T50688 C3OYQ7 9805923 IC50 = 0.068 nM T50688 CNM8S0 9806690 IC50 = 40000 nM T50688 CBJ9Q5 9807152 IC50 = 2.3 nM T50688 C68UYS 9808123 IC50 = 380 nM T50688 CH05GX 9809459 Ki < 1 nM T50688 C8Z1BK 9818983 IC50 = 8300 nM T50688 C5UOC7 9819970 IC50 = 200 nM T50688 CJ75TL 9821561 IC50 = 115 nM T50688 C19PBH 9821600 IC50 = 3.9 nM T50688 CO2Z6V 9822136 Ki = 28000 nM T50688 C4TA8N 9823909 Ki = 4 nM T50688 C4LTP2 9825687 IC50 = 23.8 nM T50688 CO73TV 9825696 IC50 = 25.3 nM T50688 C3B7WM 9825804 IC50 = 0.1 nM T50688 CLR39O 9826223 IC50 = 10 nM T50688 CFZP14 9826756 IC50 = 0.25 nM T50688 C6DLN9 9827351 IC50 = 6.1 nM T50688 CQ25XG 9827352 IC50 = 0.0058 nM T50688 C7I0XB 9827873 IC50 = 22 nM T50688 CB8GP1 9828375 IC50 = 0.31 nM T50688 CJ9HV0 9828819 IC50 = 0.16 nM T50688 C1OP9I 9828979 IC50 = 9800 nM T50688 CR8OB5 9829206 Ki = 2.3 nM T50688 CA1XU5 9842047 IC50 = 2 nM T50688 CTDP48 9843636 IC50 = 688 nM T50688 C7L0QF 9844010 IC50 = 125.89 nM T50688 C1SJR6 9844061 IC50 = 138 nM T50688 C31UCL 9844289 Ki = 30000 nM T50688 C25SWU 9844694 IC50 = 113 nM T50688 C0L7UV 9845476 IC50 = 22000 nM T50688 CPK21J 9845731 IC50 = 42 nM T50688 CZ0AS2 9846634 IC50 = 965 nM T50688 CY63LZ 9846660 IC50 = 533 nM T50688 CG0H4P 9847624 IC50 > 10000 nM T50688 C13KPA 9848051 Ki < 10000 nM T50688 CAR4I2 9849008 IC50 > 10000 nM T50688 C12AFP 9849392 IC50 = 35 nM T50688 C13OZW 9850433 IC50 = 0.78 nM T50688 CTM7V0 9851337 IC50 = 257 nM T50688 C2XD7P 9851886 IC50 > 100000 nM T50688 CCUK35 9853139 IC50 = 5 nM T50688 CR38MP 9853559 IC50 = 34700 nM T50688 CEAF74 9858710 IC50 = 32466 nM T50688 C6E3OL 9863046 Ki = 0.0465 nM T50688 C7SME4 9863277 IC50 = 110 nM T50688 CR0D9E 9864936 IC50 = 36 nM T50688 C0G1XS 9865309 IC50 = 439 nM T50688 CS4T0P 9865840 IC50 = 153 nM T50688 CZC31S 9867414 IC50 = 46 nM T50688 CR7T6A 9868824 IC50 = 105 nM T50688 CP4U2K 9869048 IC50 > 10000 nM T50688 CPKL80 9869692 IC50 > 100000 nM T50688 C2ZAK6 9870468 IC50 > 400000 nM T50688 CHC56Q 9870640 IC50 = 0.3 nM T50688 C9KN3Q 9872164 IC50 = 0.21 nM T50688 C31WAF 9872696 IC50 = 240 nM T50688 C48OAX 9872930 IC50 = 6 nM T50688 C3JA4P 9884008 IC50 = 270 nM T50688 C5EJN9 9884317 IC50 > 20000 nM T50688 C1RP4J 9884941 IC50 = 20 nM T50688 CV4T6H 9885053 IC50 > 20000 nM T50688 CJ5Z0U 9885197 IC50 = 43 nM T50688 C13WGE 9886306 IC50 > 10000 nM T50688 C1EQN3 9888685 IC50 = 104 nM T50688 C6ODX3 9888704 IC50 = 23000 nM T50688 C7B3KI 9893323 IC50 = 8 nM T50688 C49EQN 9893755 IC50 = 11 nM T50688 C6PNG8 9894403 IC50 = 3200 nM T50688 C1ZWO4 9904909 IC50 = 13 nM T50688 CNX29T 9907082 IC50 = 9 nM T50688 CMU27A 9907178 IC50 = 76 nM T50688 C2DTH6 9907685 IC50 = 1.9 nM T50688 CC6PJ4 9908437 Ki > 10000 nM T50688 CVK15W 9908440 IC50 = 15 nM T50688 C43TPN 9910543 IC50 > 10000 nM T50688 C25HTY 9910653 IC50 = 10000 nM T50688 CE34GC 9910784 IC50 = 2.7 nM T50688 CR9C5Z 9911060 Ki > 50000 nM T50688 CD7I4Y 9911639 Ki = 9000 nM T50688 CV97OQ 9912737 Ki = 0.17 nM T50688 CBZ20D 9913337 IC50 = 0.0013 nM T50688 CR13IL 9914166 IC50 > 1000 nM T50688 COT86Q 9915619 IC50 = 21 nM T50688 C69XAB 9916695 IC50 = 1300 nM T50688 CF4J2Z 9923982 IC50 > 20000 nM T50688 CUBV32 9924032 IC50 > 20000 nM T50688 CCPD70 9927009 IC50 = 1.1 nM T50688 C40MDV 9927904 IC50 = 39 nM T50688 CTNI30 9929455 IC50 = 196 nM T50688 CJPZ87 9930471 IC50 = 4360 nM T50688 CR5N6D 9931153 IC50 = 18 nM T50688 CODI28 9932234 IC50 = 0.016 nM T50688 CC42WD 9932423 IC50 = 1800 nM T50688 CT6S7L 9933202 IC50 = 6000 nM T50688 CMJ76L 9936566 IC50 = 27000 nM T50688 CP8IO3 9941178 IC50 = 10100 nM T50688 C3G5RK 9941719 IC50 = 4100 nM T50688 CUC31Q 9950075 IC50 > 50000 nM T50688 CN2Y5D 9950151 IC50 = 33 nM T50688 CLA39Q 9950422 IC50 = 600 nM T50688 C1UK7T 9953715 Ki = 36000 nM T50688 CDQ17J 9953718 IC50 = 10 nM T50688 CYG4S2 9954358 IC50 > 10000 nM T50688 C9CKS6 9956141 IC50 = 263 nM T50688 C4XK2S 9956830 IC50 = 170 nM T50688 CDU79H 9957105 IC50 = 0.59 nM T50688 CH1Y7E 9957565 IC50 = 80 nM T50688 CGP18L 9957723 IC50 = 43 nM T50688 C3VWH1 9957860 IC50 = 21.88 nM T50688 CWUC80 9958350 Ki = 128 nM T50688 C2EX4U 9972378 IC50 = 24000 nM T50688 C3PYH6 9975679 IC50 = 10000 nM T50688 C2QOL4 9978473 IC50 = 580 nM T50688 C9M2JU 9978549 IC50 = 213 nM T50688 CUIF89 9979634 IC50 = 150 nM T50688 CIXB62 9979842 IC50 > 3000 nM T50688 C9PL2H 9980010 IC50 = 740 nM T50688 C26PYH 9980810 IC50 = 59000 nM T50688 CW2ZR6 9982004 IC50 = 15 nM T50688 CXN45H 9983052 IC50 = 14000 nM T50688 CS9QB2 9983098 Ki = 3 nM T50688 CYA0W2 9983143 IC50 = 95.1 nM T50688 CPE58N 9984136 IC50 > 3000 nM T50688 CV2D0B 9984142 IC50 = 44 nM T50688 CS9VD0 9984206 IC50 = 8 nM T50688 C81DKG 9993820 IC50 = 35000 nM T50688 CN3EO0 9994930 IC50 = 5800 nM T50688 CLB29G 9996802 IC50 = 20 nM T50688 CY94QV 9999236 IC50 = 74 nM T50688 CI1HJ3 10002632 IC50 = 108 nM T50688 C6CWQ8 10003119 IC50 = 2004 nM T50688 CEJ78G 10004109 IC50 = 880 nM T50688 CV0G6H 10004443 IC50 = 18 nM T50688 C24MDH 10022569 IC50 = 3800 nM T50688 C7UZI3 10024672 IC50 = 8000 nM T50688 CBT02G 10026044 IC50 = 6610 nM T50688 CEC9V5 10026930 IC50 = 61 nM T50688 CEJ31C 10027119 IC50 = 484 nM T50688 CGT4D2 10027594 IC50 = 10882 nM T50688 CZ47BK 10027732 IC50 = 1170 nM T50688 C5CZ8A 10028351 IC50 > 10000 nM T50688 C06INP 10029120 IC50 = 37 nM T50688 CY0T9L 10030149 IC50 = 278 nM T50688 C0SU3C 10031320 IC50 = 290 nM T50688 CE2CK1 10032445 IC50 > 100000 nM T50688 CR2F8U 10043404 IC50 = 48 nM T50688 CKYE52 10044478 IC50 = 320 nM T50688 CW9O1B 10045567 IC50 = 10000 nM T50688 CPM36N 10045699 IC50 = 302 nM T50688 C6ZM5H 10047912 IC50 = 35 nM T50688 CGA89W 10049569 IC50 > 10000 nM T50688 C27XYG 10050154 IC50 = 70000 nM T50688 C86AUR 10050355 IC50 = 1100 nM T50688 CD6SV4 10050710 IC50 = 2400 nM T50688 CLS1F7 10051002 IC50 = 65.4 nM T50688 COH3U6 10052945 IC50 = 57.6 nM T50688 C89RLI 10067208 IC50 = 79 nM T50688 C40FMW 10069462 IC50 = 330 nM T50688 C2R7TW 10069591 IC50 = 780 nM T50688 CM5PL6 10069800 IC50 = 47 nM T50688 C3WZR0 10069974 IC50 = 1200 nM T50688 C7UNJ1 10071004 IC50 = 0.061 nM T50688 C25GLI 10072571 IC50 = 100 nM T50688 CFSU38 10073745 IC50 = 2 nM T50688 CK0G2T 10073952 IC50 = 350 nM T50688 CH0Y4Z 10074600 IC50 = 1470 nM T50688 C7C6FP 10074635 Ki = 1.5 nM T50688 C4AW6G 10075410 IC50 = 7 nM T50688 C6B7OI 10087503 IC50 = 18000 nM T50688 CT4O8V 10092389 IC50 = 36000 nM T50688 CO8J9N 10093461 IC50 = 158 nM T50688 C67KRY 10094447 IC50 = 54 nM T50688 CV83XM 10095387 IC50 = 240 nM T50688 CF65YE 10095540 IC50 = 5200 nM T50688 C82XUE 10095734 IC50 = 0.5 nM T50688 CLN76R 10096459 IC50 = 4050 nM T50688 CDEA39 10096654 IC50 = 4030 nM T50688 C6JLQ8 10097012 IC50 > 1000 nM T50688 C1EO7I 10098015 IC50 = 30 nM T50688 CS2A6F 10098382 IC50 = 24.4 nM T50688 C1X6MY 10099012 Ki = 110 nM T50688 CA05EG 10101088 Ki = 45 nM T50688 CESP84 10113832 IC50 > 30000 nM T50688 CWT3Y7 10136986 IC50 = 950 nM T50688 COFK25 10160125 IC50 = 20 nM T50688 CNBL36 10160126 IC50 = 34000 nM T50688 C1O0GR 10162362 IC50 = 12607 nM T50688 CX7A1Z 10164947 IC50 = 747 nM T50688 CDL31V 10165701 IC50 = 419 nM T50688 CV0G1X 10181237 IC50 = 1020 nM T50688 CO8D9C 10196873 IC50 > 10000 nM T50688 CPT2Q5 10224943 IC50 = 1400 nM T50688 C53NHL 10228662 IC50 = 8130 nM T50688 CIZ09S 10230114 IC50 = 3 nM T50688 C0M7FC 10248023 IC50 = 40 nM T50688 CJG6U3 10251891 IC50 = 23 nM T50688 CH9AD2 10252306 IC50 > 1000000 nM T50688 CM9UQ8 10252576 IC50 = 80.3 nM T50688 C7T4BQ 10252696 IC50 = 6200 nM T50688 COT17X 10254067 IC50 = 65000 nM T50688 CK8S7O 10254771 IC50 > 100000 nM T50688 CQS29V 10254830 IC50 = 45000 nM T50688 C0J5CR 10254942 IC50 = 29 nM T50688 CZ2R6D 10255598 IC50 = 3500 nM T50688 CHX06T 10255701 IC50 = 260 nM T50688 C59BFD 10256182 IC50 = 10 nM T50688 C9JOB1 10274638 IC50 = 16000 nM T50688 CD04QE 10279663 IC50 = 474 nM T50688 C7E8PX 10281105 IC50 = 0.44 nM T50688 CIF59V 10281222 IC50 = 0.18 nM T50688 C9CST0 10281487 IC50 = 18 nM T50688 CJE72C 10295656 IC50 = 35774 nM T50688 CR2YI9 10297636 IC50 = 81.9 nM T50688 CF2A5U 10317079 IC50 = 74 nM T50688 CX80NC 10318813 IC50 = 364 nM T50688 CK5LC9 10319753 IC50 = 1500 nM T50688 CB80UA 10320733 IC50 = 1900 nM T50688 C20SHE 10322151 IC50 = 3000 nM T50688 CECM40 10322684 IC50 = 18 nM T50688 CH5F6W 10322871 IC50 > 10000 nM T50688 CUZ8V6 10323749 IC50 = 4500 nM T50688 CXMC15 10325138 IC50 = 1000000 nM T50688 C7PN3T 10326558 IC50 = 4120 nM T50688 C0WZS7 10326940 IC50 = 20 nM T50688 CMP36Y 10327110 IC50 = 1.5 nM T50688 C4I2TF 10335848 IC50 = 904 nM T50688 CSO64L 10335906 IC50 = 30000 nM T50688 C14ZPK 10336754 IC50 = 2800 nM T50688 COL4X9 10340606 IC50 = 95000 nM T50688 C84KLV 10340994 IC50 = 2400 nM T50688 CYXW23 10343956 IC50 = 260 nM T50688 CR5VI0 10344187 IC50 = 1000 nM T50688 C75OLX 10344202 IC50 = 110 nM T50688 CD1C7I 10345263 IC50 = 224 nM T50688 CF18LZ 10345912 IC50 = 384 nM T50688 CJ19HI 10346506 IC50 = 36.31 nM T50688 C62KDF 10347784 Ki = 0.1 nM T50688 C1ZC2P 10348465 IC50 = 1600 nM T50688 CZPQ03 10348588 Ki = 8750 nM T50688 CM5C9S 10348589 Ki = 20 nM T50688 C39XZM 10359266 IC50 = 256 nM T50688 C2JU5Z 10359401 IC50 = 133 nM T50688 C52YXA 10363350 IC50 = 321 nM T50688 CI3AF9 10367229 IC50 = 6195 nM T50688 CQ04DG 10367832 IC50 = 36.2 nM T50688 C98AHY 10368152 IC50 = 43 nM T50688 CY1R0K 10368440 IC50 = 4362 nM T50688 C1O9DY 10369377 IC50 = 400 nM T50688 CVOY03 10369856 IC50 = 61000 nM T50688 C9THO5 10371227 IC50 = 20 nM T50688 CS24DZ 10381857 IC50 = 760 nM T50688 CK8U5J 10384651 IC50 = 64 nM T50688 CQ4H3K 10386147 IC50 = 772 nM T50688 C28BIN 10386305 IC50 = 5 nM T50688 CY51PK 10388633 IC50 = 38000 nM T50688 CZ8L0B 10389185 IC50 = 313 nM T50688 CU7V6R 10390852 IC50 = 23000 nM T50688 C7OEB8 10391124 IC50 = 0.041 nM T50688 C31WGJ 10391128 IC50 = 340 nM T50688 CC0L8M 10392074 IC50 = 4230 nM T50688 C4J3XW 10394724 Ki = 24.5 nM T50688 CL9SM7 10404377 IC50 = 100 nM T50688 C3LZ7E 10405336 IC50 = 491 nM T50688 CBL9Y6 10407528 IC50 = 290 nM T50688 C74LKV 10409937 IC50 = 1000 nM T50688 CEP9G0 10410948 IC50 = 559 nM T50688 CWH42Z 10411419 IC50 = 1000 nM T50688 CO0FY6 10411523 IC50 > 10000 nM T50688 C7B3MO 10412184 IC50 > 10000 nM T50688 CR0F1T 10412890 IC50 = 37.6 nM T50688 C7NQW0 10413380 IC50 = 4260 nM T50688 CAHU62 10413821 IC50 = 17500 nM T50688 CZ30YD 10414275 IC50 = 23.99 nM T50688 CFP6E5 10414330 IC50 = 1 nM T50688 CZ12CP 10415384 IC50 = 480 nM T50688 C2F0NO 10422987 IC50 > 100000 nM T50688 C71VHN 10426654 IC50 = 2600 nM T50688 C5VN6I 10427709 IC50 = 280 nM T50688 C4KL7O 10433389 IC50 = 600 nM T50688 CUHY62 10433896 IC50 = 27 nM T50688 C69WHT 10434168 IC50 = 500 nM T50688 C2PZQ3 10434644 IC50 = 50000 nM T50688 CTGO27 10434789 IC50 = 22000 nM T50688 CRP82B 10435346 IC50 > 10000 nM T50688 C9F2QA 10436174 IC50 = 252 nM T50688 CD8MU7 10436196 IC50 = 11200 nM T50688 C1ME0S 10436235 IC50 = 39.4 nM T50688 CT60XI 10437052 IC50 = 12000 nM T50688 C04HQK 10437073 IC50 = 32.7 nM T50688 C9KNC8 10437414 IC50 = 25000 nM T50688 CSM7T9 10437869 IC50 = 50 nM T50688 C37TNI 10439316 Ki = 143 nM T50688 C6X8SU 10449316 IC50 = 150 nM T50688 CN83LC 10449423 IC50 = 115 nM T50688 C0IA8K 10455265 IC50 = 2600 nM T50688 C6AWI9 10456038 IC50 = 7600 nM T50688 C1XTA5 10456473 IC50 > 10000 nM T50688 C6G9YM 10457584 IC50 = 187 nM T50688 C9ZN4U 10457840 IC50 = 2515 nM T50688 CX69EL 10458074 Ki = 26 nM T50688 CBR94V 10458089 IC50 = 19000 nM T50688 C6P0ZM 10458809 IC50 > 50000 nM T50688 CGW9B0 10459259 IC50 = 15600 nM T50688 CQV26D 10459311 IC50 = 2 nM T50688 C1OPH5 10459371 IC50 = 10 nM T50688 CZ7LH3 10461739 Ki = 175 nM T50688 CM2L0R 10472801 IC50 = 1240 nM T50688 C3RJ9D 10473093 IC50 = 5700 nM T50688 C0H5CG 10473844 IC50 = 500 nM T50688 CJB80U 10475325 Ki = 3.2 nM T50688 CQ0PO9 10476004 IC50 = 63 nM T50688 C7J5NX 10478278 IC50 = 12000 nM T50688 C2S0VX 10478439 IC50 = 800 nM T50688 C04EHN 10478966 IC50 = 50000 nM T50688 CZ8G3U 10479133 IC50 = 140 nM T50688 C5FX7L 10479186 IC50 = 636 nM T50688 C0NVB7 10479802 IC50 = 405 nM T50688 C0KN6P 10479916 IC50 = 4940 nM T50688 CM48CA 10480140 IC50 = 4500 nM T50688 CUT7N4 10480781 IC50 = 75900 nM T50688 C9S2RZ 10480903 IC50 = 2 nM T50688 C6IAB4 10482388 IC50 = 559 nM T50688 C9OM3L 10482416 IC50 = 13.5 nM T50688 C45MRF 10483616 IC50 > 100000 nM T50688 CH8Z5U 10484706 Ki = 125 nM T50688 CZSU97 10495925 IC50 < 100000 nM T50688 CX9CY0 10497921 IC50 = 9000 nM T50688 C57YIO 10498183 IC50 = 27 nM T50688 CIDX93 10498794 IC50 = 0.42 nM T50688 C32ENG 10498863 IC50 = 1.6 nM T50688 C7MEW6 10500045 Ki = 1200 nM T50688 C9NI6T 10500892 IC50 = 170 nM T50688 CO57MY 10501597 IC50 = 1400 nM T50688 CM0ZW9 10503055 IC50 = 250 nM T50688 CE5N7J 10504150 IC50 = 14 nM T50688 C1U8TQ 10504200 IC50 > 1000 nM T50688 C5UMV6 10504763 IC50 = 37 nM T50688 C0U6NB 10504802 IC50 = 170 nM T50688 CF24JN 10505627 IC50 = 9000 nM T50688 CWLQ37 10506080 IC50 = 7 nM T50688 CR26WA 10506313 IC50 = 390 nM T50688 CS9N1R 10506318 IC50 = 900 nM T50688 CT1FK6 10506679 IC50 = 57 nM T50688 C3W8VJ 10507104 IC50 = 39 nM T50688 CZ70VF 10507218 IC50 = 2000 nM T50688 CC58KL 10507483 IC50 = 6500 nM T50688 CXS79H 10507484 IC50 = 11000 nM T50688 CKT5B3 10521604 IC50 = 850 nM T50688 CPI81M 10521872 IC50 = 0.12 nM T50688 C3ZK9B 10521873 IC50 = 5 nM T50688 CHF70E 10523877 Ki = 1750 nM T50688 C2HV8Y 10524492 IC50 = 0.13 nM T50688 C17VLR 10525508 IC50 = 78 nM T50688 C2KW1M 10525856 IC50 = 0.81 nM T50688 CW37AZ 10526036 IC50 > 1000 nM T50688 C4VN0A 10526120 IC50 = 21 nM T50688 C7DQU0 10526203 Ki > 50000 nM T50688 CEU48D 10526463 IC50 = 180 nM T50688 CA7Q1M 10526820 IC50 = 340 nM T50688 COY51D 10527580 IC50 = 0.14 nM T50688 CD6T3L 10527653 IC50 > 1000 nM T50688 C43BPT 10527958 IC50 = 12 nM T50688 C0D6XG 10528000 IC50 = 6000 nM T50688 C4P5VR 10528032 IC50 = 4200 nM T50688 C16HLY 10528334 IC50 = 6000 nM T50688 CGE0P3 10528399 Ki = 540 nM T50688 C2AX9H 10528472 IC50 = 32 nM T50688 CV06QK 10528788 IC50 = 300 nM T50688 C0T5IM 10529317 IC50 = 6300 nM T50688 CM4Z9C 10529546 IC50 = 1000 nM T50688 CC9GJ8 10529586 IC50 = 24 nM T50688 C0G5VX 10529678 IC50 = 95 nM T50688 CUY9Q0 10529865 IC50 > 10000 nM T50688 C3FG5K 10530186 IC50 = 9 nM T50688 CQ8JT1 10530357 IC50 = 4.3 nM T50688 C61HVA 10530613 IC50 = 260 nM T50688 CG1H4C 10531830 IC50 = 27.3 nM T50688 C2L1PJ 10531967 IC50 = 1600 nM T50688 CF0CS2 10541651 IC50 = 18000 nM T50688 CU95VC 10544052 IC50 = 16000 nM T50688 CPC51L 10544691 IC50 = 46000 nM T50688 C1WA0R 10545460 IC50 = 9900 nM T50688 CD1Y5N 10546320 IC50 = 440 nM T50688 CBS2F4 10548981 IC50 > 1000 nM T50688 CWA51X 10549838 IC50 = 3 nM T50688 CY4QG2 10549931 IC50 = 0.92 nM T50688 C3ST9M 10549992 IC50 = 130 nM T50688 C1SJN7 10551324 IC50 = 96 nM T50688 C8Y3PH 10551831 IC50 = 125 nM T50688 CBJ70D 10551898 IC50 = 15 nM T50688 CEO2N5 10552647 IC50 = 930 nM T50688 CR6TH2 10553451 IC50 = 2630 nM T50688 C7BLP8 10553605 IC50 = 180 nM T50688 C1OP8Z 10554323 IC50 = 45 nM T50688 CZD20R 10555279 IC50 = 3100 nM T50688 CAFZ87 10555310 IC50 = 260 nM T50688 C1S5KM 10555762 IC50 = 31.3 nM T50688 CPX62H 10567014 IC50 = 630 nM T50688 C02LOP 10569012 IC50 = 260 nM T50688 CTKA09 10569078 IC50 = 1200 nM T50688 C45UKM 10569143 IC50 = 12000 nM T50688 C63AQL 10569459 IC50 = 4100 nM T50688 C7PIF3 10569520 IC50 = 7400 nM T50688 C5K6LD 10570053 IC50 = 190 nM T50688 CR0WY1 10570641 IC50 = 12000 nM T50688 C6ST5A 10570949 IC50 = 500 nM T50688 CU01OT 10572765 Ki = 290 nM T50688 CI4CM8 10573992 IC50 = 170 nM T50688 C95HGK 10574096 IC50 = 130 nM T50688 CAWF40 10574237 Ki > 100000 nM T50688 CDZR27 10574289 IC50 = 360 nM T50688 CMN41A 10574669 IC50 = 7.2 nM T50688 CC9M4O 10574710 IC50 = 0.2 nM T50688 C1K8IY 10574717 IC50 = 85 nM T50688 COA4T1 10574792 IC50 = 8.1 nM T50688 C75XGA 10574888 IC50 = 2500 nM T50688 C73VFG 10574923 IC50 = 20 nM T50688 C01GQV 10575330 IC50 = 36 nM T50688 C47OMC 10575410 IC50 = 5000 nM T50688 C5P1NG 10575581 IC50 = 73 nM T50688 CI35XW 10576070 Ki = 80 nM T50688 C6NM7V 10576167 IC50 = 69 nM T50688 CXZP31 10576168 IC50 = 67 nM T50688 CB67ER 10576733 IC50 = 13000 nM T50688 CV3QL4 10577095 IC50 = 1.8 nM T50688 CX1K0N 10577150 IC50 = 21 nM T50688 CKP4H6 10577279 IC50 = 1.5 nM T50688 CJ3T2Q 10577940 IC50 = 12 nM T50688 CU75WP 10578810 IC50 = 81 nM T50688 CZ9VX1 10579340 IC50 = 21.3 nM T50688 C0U1CG 10582643 IC50 > 10000 nM T50688 CWG26D 10591778 IC50 = 44000 nM T50688 CQ5LE9 10592825 IC50 = 10000 nM T50688 CF15AC 10593246 IC50 = 77000 nM T50688 CLA3Q4 10595524 IC50 = 160 nM T50688 CS15AP 10596310 IC50 = 16000 nM T50688 CZ9ES6 10596311 IC50 = 25300 nM T50688 CDK10F 10597871 IC50 = 40 nM T50688 CKS6B5 10598109 IC50 = 60 nM T50688 C8TQ3C 10598184 IC50 = 42 nM T50688 CDM3L1 10598267 IC50 = 2200 nM T50688 CC4AS1 10598742 IC50 = 0.13 nM T50688 CM38KV 10598938 IC50 = 1030 nM T50688 C9SM8R 10599499 IC50 = 230 nM T50688 C4I2EJ 10599577 IC50 = 88 nM T50688 CE7DI4 10600322 IC50 = 47 nM T50688 CNO98S 10600933 IC50 = 0.34 nM T50688 CJ16VT 10601205 IC50 = 0.52 nM T50688 C6WK7Z 10601297 IC50 = 3 nM T50688 CC52PM 10601502 IC50 = 1.8 nM T50688 CI09PZ 10601521 IC50 = 32 nM T50688 CSZ1C6 10601709 IC50 = 3.6 nM T50688 CA04QH 10601955 IC50 = 0.85 nM T50688 CLA7F4 10602103 IC50 = 11 nM T50688 CA0NM6 10602590 IC50 = 26 nM T50688 C39IPX 10603319 IC50 = 12 nM T50688 C07MCW 10603422 IC50 = 470 nM T50688 CAW3U8 10603619 IC50 = 11 nM T50688 C0EU7G 10603811 IC50 = 34.7 nM T50688 CPVM74 10604005 IC50 = 2 nM T50688 CDXB14 10606654 IC50 > 1000 nM T50688 CJ49TW 10615755 IC50 = 1100 nM T50688 CY86JI 10617432 IC50 > 100000 nM T50688 CNB89K 10620252 IC50 > 10000 nM T50688 C1V9UK 10620480 IC50 = 0.26 nM T50688 C7N8UQ 10621705 IC50 > 1000 nM T50688 CRFI52 10622095 IC50 = 0.1 nM T50688 CB7X1D 10622197 IC50 = 500 nM T50688 CUME64 10622650 IC50 = 0.21 nM T50688 CT9U1I 10622651 IC50 = 2810 nM T50688 CZ1D7P 10622934 IC50 = 0.22 nM T50688 CIL20A 10623555 IC50 = 31 nM T50688 C35QBJ 10623736 IC50 = 350 nM T50688 C1VC0O 10624584 IC50 = 3.8 nM T50688 C5FGS8 10624764 Ki = 800 nM T50688 CLR06I 10626114 IC50 = 57 nM T50688 CMQA47 10626357 IC50 = 5.1 nM T50688 C08FHO 10627561 IC50 = 3410 nM T50688 CUBJ20 10628601 IC50 = 67 nM T50688 CA03HK 10639257 IC50 = 55000 nM T50688 C0CFP3 10639900 IC50 = 5000 nM T50688 CBZ8U6 10641657 IC50 = 4200 nM T50688 CF8CK1 10644680 IC50 = 0.58 nM T50688 CLV5I7 10645125 IC50 = 300 nM T50688 C1TKQ4 10645607 IC50 = 8000 nM T50688 CMB93Z 10645847 Ki > 50000 nM T50688 CS5PN3 10647720 IC50 > 1000 nM T50688 CM54PX 10647971 IC50 > 1000 nM T50688 C0EFS9 10648519 IC50 = 85000 nM T50688 C5ABX8 10648597 Ki = 26 nM T50688 CX98VN 10648960 IC50 = 1500 nM T50688 CY38BT 10649923 IC50 = 6500 nM T50688 CHV18W 10650104 IC50 = 74 nM T50688 C91EXP 10650216 IC50 = 5.4 nM T50688 CI3E1K 10650223 IC50 = 44 nM T50688 CIW40L 10650245 IC50 = 5.8 nM T50688 CW5KO9 10650595 IC50 = 41000 nM T50688 C4QO9H 10651012 IC50 = 130 nM T50688 CXQ5B4 10663504 IC50 = 23000 nM T50688 CI0K7L 10665207 IC50 = 26700 nM T50688 CD82QM 10666108 IC50 = 27000 nM T50688 C5OQJ8 10666236 IC50 = 1800 nM T50688 C8SH0G 10667601 IC50 = 4000 nM T50688 CP18RM 10669069 IC50 = 460 nM T50688 C6V4RM 10669472 IC50 = 2100 nM T50688 C0F7QU 10669861 IC50 = 10000 nM T50688 C3TJ1R 10669871 IC50 = 0.15 nM T50688 CUIE47 10670418 IC50 = 20 nM T50688 CU13QF 10670421 IC50 = 100 nM T50688 C8QTJ0 10670464 IC50 = 78 nM T50688 C7UA2O 10671221 IC50 = 230 nM T50688 CPMD78 10671690 IC50 = 41 nM T50688 CK87TJ 10672605 IC50 > 10000 nM T50688 C8O5EP 10672609 IC50 = 61 nM T50688 CMB4O8 10673127 IC50 > 10000 nM T50688 CVX5L8 10673284 IC50 = 5000 nM T50688 C5C4KF 10673305 IC50 = 34 nM T50688 C4OU1Z 10673351 IC50 = 67 nM T50688 C1K4VA 10673587 IC50 = 290 nM T50688 C9AO8W 10673593 IC50 = 15 nM T50688 CNZ52W 10674738 IC50 = 4400 nM T50688 CN07MA 10675175 IC50 = 47.3 nM T50688 C5CO8D 10675509 IC50 = 64 nM T50688 CY10JG 10678157 IC50 > 1000 nM T50688 CMV21P 10678163 IC50 > 1000 nM T50688 C6R4MV 10678165 IC50 > 10000 nM T50688 CO35RT 10686097 IC50 = 28000 nM T50688 CF73WA 10687020 IC50 = 60 nM T50688 CG68IP 10688817 IC50 = 310 nM T50688 CL61KC 10689869 IC50 = 140 nM T50688 CDVJ25 10690277 IC50 = 410 nM T50688 CNW32D 10690754 IC50 = 1800 nM T50688 C6U0EH 10691302 IC50 > 10000 nM T50688 CM4I0K 10692763 Ki = 52000 nM T50688 CBJ5U8 10693286 IC50 = 1.7 nM T50688 CX6R5Z 10693378 IC50 = 1 nM T50688 CIP7S4 10693570 IC50 = 2.6 nM T50688 C7F6CR 10693833 Ki = 2.5 nM T50688 CTV09E 10695326 Ki = 19 nM T50688 C6G5SF 10696089 IC50 = 50 nM T50688 COE2C0 10696268 Ki = 2 nM T50688 CT08OR 10696562 IC50 = 570 nM T50688 CLYC49 10697230 IC50 = 10 nM T50688 CX26BU 10697338 IC50 > 10000 nM T50688 C3SF8N 10697605 IC50 = 32000 nM T50688 CFG8O6 10698251 IC50 = 400 nM T50688 CYV8S2 10698274 IC50 = 66 nM T50688 CHL29X 10698729 IC50 = 10 nM T50688 C98TZX 10699307 IC50 = 1370 nM T50688 CWP46I 10710664 IC50 = 36600 nM T50688 CBH0X7 10710665 IC50 = 38200 nM T50688 CRP1Q5 10711631 IC50 = 18000 nM T50688 C57MHS 10711633 IC50 = 11000 nM T50688 CK6OM7 10711689 IC50 = 91 nM T50688 CXE5V7 10712480 IC50 = 43700 nM T50688 CU90KW 10714203 Ki = 560 nM T50688 CIMF59 10715577 Ki > 50000 nM T50688 C4D2UE 10716904 IC50 = 138 nM T50688 C3CG9M 10717156 IC50 = 40 nM T50688 C9JRQ6 10717165 IC50 = 180 nM T50688 C30YKM 10718276 IC50 = 34000 nM T50688 CPZ2J1 10718421 IC50 = 110 nM T50688 CI3F1Z 10719036 IC50 = 0.18 nM T50688 CJ9WY6 10719690 Ki = 14900 nM T50688 C9T4FM 10720025 IC50 = 18 nM T50688 CB2JR1 10720397 IC50 = 180 nM T50688 CY40LK 10720760 IC50 = 850 nM T50688 C4LY7B 10720773 IC50 = 0.66 nM T50688 CWM1H4 10721018 IC50 = 4 nM T50688 CYM68T 10721510 IC50 = 57 nM T50688 CRD6A2 10734460 IC50 = 19000 nM T50688 C4DL1X 10735250 IC50 = 1100 nM T50688 CD8QH7 10736235 IC50 = 7500 nM T50688 C7ISZ3 10737628 Ki = 1500 nM T50688 CMCP54 10737883 IC50 = 40 nM T50688 CO9EB6 10739023 IC50 = 50 nM T50688 C3JG8M 10739084 IC50 = 0.16 nM T50688 CFEW14 10740150 IC50 = 50000 nM T50688 CY40JW 10741088 IC50 = 21 nM T50688 C0WB5V 10741543 IC50 = 5000 nM T50688 C32HFP 10741551 IC50 = 65 nM T50688 CTF43Q 10741717 IC50 = 3 nM T50688 CW1V6I 10741784 IC50 = 180 nM T50688 C5F6IQ 10742630 IC50 = 210 nM T50688 CQ43HK 10743381 IC50 = 2 nM T50688 CA5BC6 10743635 IC50 = 10000 nM T50688 C3EY2G 10744029 IC50 = 32 nM T50688 CQN7C5 10744439 IC50 = 5.3 nM T50688 CWTH73 10744841 IC50 = 36 nM T50688 C72AXW 10744879 IC50 = 3100 nM T50688 CPW19S 10744934 IC50 = 7800 nM T50688 C0XJY2 10745059 IC50 = 13 nM T50688 CS7YL2 10745179 IC50 = 190 nM T50688 C5N0JC 10745304 IC50 = 5000 nM T50688 CE0DW6 10745412 IC50 = 3.8 nM T50688 C2YL0X 10745414 IC50 = 2.7 nM T50688 CDHZ35 10745638 IC50 = 770 nM T50688 CPQ9N3 10746038 IC50 = 65 nM T50688 CTZG52 10746372 IC50 = 74 nM T50688 CI6W7O 10747110 IC50 = 22 nM T50688 C5GA7Z 10747212 IC50 = 11 nM T50688 CJ6EY5 10760011 IC50 = 48000 nM T50688 C2J5DF 10760306 IC50 = 14000 nM T50688 C2UVP6 10760519 IC50 = 0.073 nM T50688 CWA45B 10762449 IC50 = 14000 nM T50688 CU79QS 10764595 IC50 = 2.5 nM T50688 CD5BH1 10765679 IC50 = 0.75 nM T50688 C0BW1Q 10765828 IC50 = 90 nM T50688 C36RIG 10765872 IC50 = 50000 nM T50688 CC47BU 10765873 IC50 = 1000 nM T50688 C65WOR 10766035 IC50 = 1000 nM T50688 C0Q8ET 10766137 IC50 = 20 nM T50688 CC06BN 10766594 IC50 = 31 nM T50688 C4XFU2 10767331 IC50 = 3000 nM T50688 CUB46C 10767352 IC50 = 600 nM T50688 CRK0M2 10767647 IC50 = 2 nM T50688 CL1XE6 10767757 IC50 = 10 nM T50688 CO15MH 10769104 IC50 = 5000 nM T50688 CH35PG 10780340 IC50 > 100000 nM T50688 CD38LF 10780686 IC50 = 48000 nM T50688 CG1B9U 10781733 IC50 = 2300 nM T50688 CDZM40 10781802 IC50 = 60 nM T50688 CL9M4R 10783789 IC50 = 6000 nM T50688 CJBT94 10784172 IC50 = 5 nM T50688 C7QDL1 10786753 IC50 = 0.13 nM T50688 CJE7P8 10788151 IC50 = 330 nM T50688 C0Z5PU 10788266 IC50 = 21000 nM T50688 CBJK78 10788353 IC50 = 630 nM T50688 CR2Y3H 10788405 Ki = 8 nM T50688 CYC0D7 10788947 IC50 = 1 nM T50688 CU6M5W 10788997 IC50 = 250000 nM T50688 C5B6MC 10789118 IC50 = 13 nM T50688 C25HXT 10789240 IC50 = 0.24 nM T50688 CRLY08 10790058 IC50 > 1000 nM T50688 CL07VH 10790223 IC50 = 250 nM T50688 CL48DH 10790594 IC50 = 0.65 nM T50688 CIMC29 10790917 IC50 = 55 nM T50688 CRME39 10791865 IC50 > 10000 nM T50688 CD60VX 10791985 IC50 = 7 nM T50688 CGI2S3 10792202 IC50 = 83 nM T50688 C0IFV7 10792261 IC50 = 13 nM T50688 CKU3Z4 10792272 IC50 = 570 nM T50688 C90EQR 10793103 IC50 = 4000 nM T50688 C9L4KF 10793351 IC50 = 790 nM T50688 CG47UL 10793849 IC50 = 72 nM T50688 C5YSV2 10794013 IC50 = 5.6 nM T50688 CQE3T7 10794762 IC50 = 96 nM T50688 C56FMJ 10807406 IC50 = 340 nM T50688 C9Z1JU 10807527 IC50 = 54 nM T50688 CE80DB 10807712 IC50 = 290 nM T50688 CG70RV 10808878 IC50 = 3 nM T50688 CRJ80X 10808969 IC50 = 6000 nM T50688 CR2SG6 10809369 IC50 = 250 nM T50688 CKW54J 10810465 IC50 = 65 nM T50688 CANY49 10810509 IC50 = 594 nM T50688 CS87IC 10810880 IC50 = 6300 nM T50688 CG5Y0D 10811208 IC50 = 163 nM T50688 C5GU3F 10811614 IC50 = 10000 nM T50688 C0GAW3 10811724 IC50 = 46 nM T50688 C1EI3C 10811745 IC50 = 590 nM T50688 C2E5AI 10813353 IC50 = 18 nM T50688 C6AV1O 10813355 IC50 = 0.89 nM T50688 C0BO1X 10813883 Ki = 750 nM T50688 C86QIK 10814015 IC50 = 68 nM T50688 CQSR19 10814133 IC50 = 1600 nM T50688 CKHJ63 10814581 IC50 = 55 nM T50688 CXQD50 10814626 IC50 = 35 nM T50688 CL35GT 10815092 IC50 = 160 nM T50688 CZA18Q 10815853 IC50 = 36 nM T50688 CNG0H1 10816131 IC50 > 100000 nM T50688 C8X6GV 10816353 IC50 = 8.6 nM T50688 CVL1Q5 10816922 IC50 = 22.3 nM T50688 CXY5H4 10817117 IC50 = 8 nM T50688 CL5M9B 10817315 IC50 = 363 nM T50688 CC79QZ 10829524 IC50 = 64000 nM T50688 C7NLW3 10830476 IC50 = 870 nM T50688 CI7HF0 10830837 IC50 = 47000 nM T50688 C9LZ8N 10830937 IC50 = 30 nM T50688 C7QS2L 10831902 IC50 = 5800 nM T50688 CA8X9M 10831903 IC50 = 4000 nM T50688 CGRC85 10832778 IC50 = 600 nM T50688 CAWT74 10833338 IC50 = 210 nM T50688 CYBU67 10837146 IC50 = 360 nM T50688 CCW4P0 10838744 IC50 = 30000 nM T50688 CVX39A 10838945 IC50 = 0.21 nM T50688 C65XRV 10839051 IC50 = 0.37 nM T50688 C7I6UV 10839864 IC50 = 3.8 nM T50688 CSK2Z4 10839940 IC50 = 5 nM T50688 C06QAI 10839976 IC50 > 100000 nM T50688 CKN51D 10840512 IC50 = 11 nM T50688 CTJ61U 10840969 IC50 = 36000 nM T50688 CY9DP7 10841676 IC50 = 21 nM T50688 C7EB4Y 10844291 IC50 > 1000 nM T50688 C9XK7J 10844292 IC50 = 1000 nM T50688 C1OFW6 10850199 IC50 = 48000 nM T50688 CMU8D1 10853893 IC50 > 100000 nM T50688 CIV0X1 10961560 IC50 = 2900 nM T50688 C08BCF 10993678 IC50 = 7300 nM T50688 CDK7W9 10994476 IC50 > 10000 nM T50688 CTW0P5 11102917 IC50 > 10000 nM T50688 C79OJR 11133736 IC50 = 580 nM T50688 C1S0PM 11169785 Ki = 206 nM T50688 CBO8Q0 11181082 Ki = 6840 nM T50688 CXEH75 11187899 IC50 = 733 nM T50688 CQF31D 11190947 Ki = 973 nM T50688 C2JZ6C 11192964 Ki = 7300 nM T50688 CJU1K7 11200734 IC50 > 10000 nM T50688 C5SH1R 11227896 Ki = 3660 nM T50688 CN74QM 11234552 IC50 = 660 nM T50688 CQG0I1 11234588 IC50 = 350 nM T50688 C4HFS8 11234619 IC50 = 17 nM T50688 C8A5RL 11237915 Ki = 3940 nM T50688 C83HIU 11246220 IC50 = 1610 nM T50688 CR2JN6 11246637 IC50 = 329 nM T50688 CPQ2H7 11246987 IC50 = 841 nM T50688 C5JXU9 11257283 IC50 = 5183 nM T50688 CDN62X 11269177 IC50 = 4 nM T50688 CY1LH0 11281059 IC50 = 68 nM T50688 C98HYU 11284340 IC50 = 1 nM T50688 CSH76U 11284767 IC50 = 24630 nM T50688 CWN52M 11292505 IC50 = 730 nM T50688 CVW45L 11292510 IC50 = 5 nM T50688 CA7EI1 11304190 IC50 = 212 nM T50688 CVQ9A3 11304592 IC50 = 3600 nM T50688 C7HTY1 11307791 IC50 = 2 nM T50688 C51AZT 11315587 IC50 = 6490 nM T50688 C82ZFG 11337742 IC50 = 5700 nM T50688 C7VDO8 11372991 IC50 = 21 nM T50688 CZJ15G 11374651 IC50 = 90 nM T50688 CZ5E4X 11374986 IC50 = 20 nM T50688 CTS8G9 11384491 IC50 = 222 nM T50688 CV1NT6 11386324 IC50 = 120 nM T50688 C45EBU 11394236 IC50 = 12500 nM T50688 C4KU1F 11395891 IC50 = 700 nM T50688 CZO3H7 11399588 IC50 = 9000 nM T50688 CL8AO4 11406569 IC50 = 751 nM T50688 CS4PY1 11406925 IC50 = 4100 nM T50688 CNP04F 11410732 IC50 = 16 nM T50688 CVI7S8 11441000 IC50 = 410 nM T50688 CE6FI4 11452378 IC50 = 1020 nM T50688 C9L2OX 11452690 IC50 > 10000 nM T50688 CEWT48 11452816 Ki = 4.2 nM T50688 CJCF34 11486406 IC50 = 3400 nM T50688 CDIR54 11486773 IC50 > 10000 nM T50688 CZ8I5T 11489856 IC50 = 5 nM T50688 C50FQZ 11489885 IC50 = 1640 nM T50688 C5NEM0 11546965 IC50 = 168 nM T50688 CFZ2O9 11613998 IC50 > 50000 nM T50688 CGU84F 11721315 IC50 > 50000 nM T50688 C2ONX6 11721442 IC50 = 8000 nM T50688 CLHR18 11723405 IC50 > 10000 nM T50688 CO7K6Z 11740268 IC50 = 105 nM T50688 CF9IT7 11740665 IC50 = 3 nM T50688 CUW59R 11741589 IC50 = 14000 nM T50688 CY35MP 11742524 IC50 = 26000 nM T50688 C01BWL 11742781 IC50 = 35 nM T50688 C7GV2M 11743323 IC50 = 29 nM T50688 C9CX0F 11743586 IC50 = 101 nM T50688 CE5H7K 11744415 IC50 = 11200 nM T50688 CIO0X8 11744424 IC50 = 300 nM T50688 CS1Q9P 11744536 IC50 > 10000 nM T50688 CZ9GM1 11749950 IC50 = 112 nM T50688 CR7NP5 11751578 IC50 = 25 nM T50688 C2KZ5U 11752405 IC50 = 5 nM T50688 CBS24R 11754911 IC50 = 3 nM T50688 CV63YK 11755157 IC50 = 29 nM T50688 CMY21B 11756777 IC50 = 65 nM T50688 CPXI40 11757187 IC50 > 3000 nM T50688 C3DCM0 11757316 IC50 = 1000000 nM T50688 CEN37T 11757623 IC50 = 220 nM T50688 C8MFU9 11772736 IC50 = 7400 nM T50688 CB5MA7 11791726 IC50 = 9800 nM T50688 C8S1AR 11791783 IC50 = 760 nM T50688 C4H6KF 11791858 IC50 = 39000 nM T50688 C39KJR 11792525 IC50 = 3.5 nM T50688 C98GJL 11792811 IC50 = 48 nM T50688 C7PY0U 11793130 IC50 = 4000 nM T50688 CV51NX 11796444 IC50 = 1350 nM T50688 CPKC53 11797034 IC50 = 47 nM T50688 CA1FD8 11797035 IC50 = 27 nM T50688 C9KVR6 11797667 IC50 = 200 nM T50688 C5GTQ0 11798113 IC50 = 200 nM T50688 CFL9C4 11799328 IC50 = 3000 nM T50688 CHIN14 11799438 IC50 = 51 nM T50688 CT4D1K 11799915 IC50 > 100000 nM T50688 C4U1TD 11800065 IC50 = 78000 nM T50688 CZ06CB 11800170 IC50 = 600 nM T50688 C2BC6I 11800172 IC50 = 11 nM T50688 C4Z5HL 11800506 IC50 = 23 nM T50688 CW73UB 11800522 IC50 = 14 nM T50688 CD0GH5 11800573 IC50 > 100000 nM T50688 COT19X 11800615 IC50 = 410 nM T50688 CYC1X9 11800819 IC50 = 8100 nM T50688 C30JTG 11801283 IC50 = 5.7 nM T50688 CBF42H 11802695 IC50 = 22 nM T50688 C7EKZ0 11975699 Ki = 7.1 nM T50688 C1E9BA 12096120 IC50 = 660 nM T50688 CNA3W7 14563588 IC50 = 20000 nM T50688 CB2TD1 14796453 IC50 = 2300 nM T50688 C04GKV 15030977 IC50 = 27000 nM T50688 CV0AL8 15088298 IC50 > 200000 nM T50688 C3U8TD 15088299 IC50 = 138000 nM T50688 CDP35E 15088300 Ki = 14500 nM T50688 CKGL39 15088301 IC50 = 113000 nM T50688 C6BDE1 15088302 IC50 > 200000 nM T50688 CMK62Y 15088303 IC50 > 200000 nM T50688 C7ZOQ1 15088304 IC50 > 200000 nM T50688 C2DSH8 15088306 IC50 > 200000 nM T50688 CBL38Q 15088307 IC50 > 200000 nM T50688 CC34KU 15088308 IC50 > 200000 nM T50688 CR9ZP3 15088309 IC50 > 200000 nM T50688 CR5N7E 15088310 IC50 = 97000 nM T50688 CI69AO 15088312 IC50 > 200000 nM T50688 CNIV75 15088313 Ki < 10000 nM T50688 C6JVF0 15088314 IC50 = 102000 nM T50688 C17RXP 15088315 Ki = 4200 nM T50688 CV2UN6 15088316 IC50 > 200000 nM T50688 CGS1Y3 15088321 Ki = 3000 nM T50688 CW54MQ 15088322 Ki = 720 nM T50688 CCR3J9 15088323 Ki = 720 nM T50688 COR10Z 15088329 IC50 = 370 nM T50688 C9O8TU 15223439 IC50 = 122 nM T50688 CI7C9X 15223440 IC50 = 50 nM T50688 CP9S4I 15233759 IC50 = 170 nM T50688 CSF4Y8 15295775 IC50 = 5000 nM T50688 C69FBX 15297021 IC50 = 4.2 nM T50688 CVD8Z5 15337543 IC50 = 0.09 nM T50688 CAJ1P8 15337548 IC50 = 0.13 nM T50688 C9ZL2Y 15380364 IC50 = 125 nM T50688 C9N0XP 15428414 IC50 = 8 nM T50688 CR2MA3 15432278 IC50 = 1090 nM T50688 CMZN94 15483869 IC50 = 40 nM T50688 C7DT2P 15483870 IC50 = 24 nM T50688 C0WJ7R 15483871 IC50 = 7 nM T50688 CMES74 15486068 Ki = 30000 nM T50688 C1V8GD 15488825 Ki = 1.5 nM T50688 C2YG3M 15491369 Ki = 2300 nM T50688 COEP73 15491370 Ki = 20000 nM T50688 CZ2R8G 15491452 IC50 = 1300 nM T50688 CN0LX5 15491453 IC50 = 780 nM T50688 C3VOW7 15491454 IC50 = 460 nM T50688 CZX58V 15516067 Ki > 50000 nM T50688 CZBP40 15545291 IC50 = 11 nM T50688 CJGB65 15545292 IC50 = 72 nM T50688 C6WGZ9 15545293 IC50 = 610 nM T50688 CU60GO 15545294 IC50 = 71 nM T50688 CS81PK 15545295 IC50 = 26 nM T50688 C3OPX2 15547267 IC50 = 210 nM T50688 CZ48KQ 15838053 IC50 = 10 nM T50688 CDVB07 15850631 IC50 = 45 nM T50688 CG9FV3 15850632 IC50 = 2800 nM T50688 CKPV73 15850737 IC50 = 55 nM T50688 CM79QV 15850743 IC50 = 110 nM T50688 CM8G3S 15859412 IC50 > 10000 nM T50688 CW8LN2 15859413 IC50 = 2450 nM T50688 CT1DI8 15859414 IC50 = 2800 nM T50688 C95OGC 15859418 IC50 = 80 nM T50688 CEC41O 15859419 IC50 = 925 nM T50688 CFJ08N 15859420 IC50 = 235 nM T50688 CUQ9A2 15859421 IC50 = 55 nM T50688 C56IZT 15859422 IC50 = 9 nM T50688 CE6FO4 15859423 IC50 > 10000 nM T50688 C1VMK9 15859424 IC50 = 1000 nM T50688 C2B8GR 15887956 IC50 = 3 nM T50688 CKPY93 15887958 IC50 = 9 nM T50688 C8QO3Z 15887960 IC50 = 600 nM T50688 C8QIB4 15888084 Ki > 30000 nM T50688 CUY2F9 15931145 Ki = 1900 nM T50688 C7A0NY 15931147 IC50 > 200000 nM T50688 C9LSV8 16211712 Ki > 1000000 nM T50688 CTGC60 16678135 IC50 = 2300 nM T50688 CU8YQ3 16756502 IC50 = 7.7 nM T50688 C0KW3V 16756505 IC50 > 50000 nM T50688 C04JOX 16756621 IC50 = 50000 nM T50688 C4CU7T 16756622 IC50 > 50000 nM T50688 CFH96E 16756623 IC50 > 50000 nM T50688 CB15RX 16756849 IC50 = 12000 nM T50688 CM18ZN 16756955 IC50 > 50000 nM T50688 CL38IU 16756956 IC50 = 11000 nM T50688 CW5P8L 16756957 IC50 > 50000 nM T50688 CRWZ62 17788068 IC50 = 2700 nM T50688 C2DN9B 18394355 Ki > 50000 nM T50688 CAOR56 18660413 IC50 = 25000 nM T50688 C2HD8G 18967498 IC50 = 31000 nM T50688 C3T0QV 19034178 IC50 = 330000 nM T50688 C0O6XT 19076730 IC50 = 4810 nM T50688 C9G7ZK 19697937 IC50 = 0.098 nM T50688 C8SCL4 19757280 IC50 = 4880 nM T50688 CHV3L9 19757296 IC50 = 5880 nM T50688 CJ4L3C 19757333 IC50 = 4720 nM T50688 CW4IN3 19757343 IC50 = 2870 nM T50688 CY19FN 19962234 IC50 = 46 nM T50688 CXLO94 20587795 IC50 = 255 nM T50688 C7FR8G 20639626 IC50 = 28 nM T50688 CW64DV 20666951 IC50 = 21900 nM T50688 C85SOV 20666970 IC50 = 54 nM T50688 C61WDP 20666971 IC50 = 128 nM T50688 CX52NV 20666990 IC50 = 148 nM T50688 CVJ8N2 20667011 IC50 = 253 nM T50688 CMV17G 20667012 IC50 = 172 nM T50688 CQ8ME6 20667015 IC50 = 22 nM T50688 CR2X4L 20694723 IC50 = 4.2 nM T50688 CE57KZ 20694724 IC50 = 0.057 nM T50688 C6VZA8 20709789 IC50 > 10000 nM T50688 CEI27V 21053920 IC50 > 10000 nM T50688 C3TR2D 21191396 IC50 = 285 nM T50688 CE5Z3R 21191398 IC50 = 57 nM T50688 CGI19E 21191399 IC50 = 14.3 nM T50688 CN1Q0M 21191405 IC50 = 1000 nM T50688 C3GK7N 21191409 IC50 = 93 nM T50688 CQJ5Z3 21191417 IC50 = 3190 nM T50688 CU4FN2 21191441 IC50 = 4710 nM T50688 CM96YE 21191461 IC50 = 12.5 nM T50688 C7XYV3 21191470 IC50 = 6 nM T50688 C6X9US 21465966 IC50 = 80 nM T50688 CA10BL 21465982 IC50 = 31 nM T50688 CUJS70 21699778 IC50 > 10000 nM T50688 C2N6QA 21927945 IC50 = 9298 nM T50688 CT6N9S 22094645 IC50 = 1.2 nM T50688 CMS31G 22098946 IC50 = 1830 nM T50688 CE5G2I 22098949 IC50 = 2170 nM T50688 C2U1YQ 22098952 IC50 = 8270 nM T50688 CEU65M 22098953 IC50 = 670 nM T50688 CO4JK1 22098959 IC50 = 817 nM T50688 CN1Q2O 22098975 IC50 = 97 nM T50688 C94AUL 22098977 IC50 = 14.1 nM T50688 C7T2YX 22402471 IC50 = 2300000 nM T50688 CP2DW6 22451718 Ki = 1.9 nM T50688 CAD90V 22451721 Ki = 1.5 nM T50688 CG6FE5 22451739 Ki = 2 nM T50688 CJRA54 22451788 Ki = 22500 nM T50688 CP47JN 22451902 Ki = 4.7 nM T50688 CXVB03 22594242 IC50 = 110 nM T50688 CDJH42 22594251 IC50 = 1495 nM T50688 CPF73W 22594331 IC50 > 100000 nM T50688 CHR03I 22594351 IC50 = 1700 nM T50688 CFL7X5 22594355 IC50 = 552 nM T50688 CHVR74 22611774 IC50 = 200 nM T50688 CVM5Q1 22611776 IC50 > 100 nM T50688 C5LH4U 22611792 IC50 = 3 nM T50688 C2WR9E 22611889 IC50 > 100 nM T50688 C4V7BI 22645287 IC50 = 10 nM T50688 CB43DX 22866013 IC50 = 1.1 nM T50688 CFG40R 22975644 IC50 = 15000 nM T50688 C0MNQ9 23286727 IC50 = 47 nM T50688 CR6T1J 23297694 Ki = 1 nM T50688 CXZD95 23297711 Ki = 2 nM T50688 CWKA89 23297715 Ki = 1.7 nM T50688 CG7YV4 23297719 Ki = 1.5 nM T50688 CMG08E 23297721 Ki = 2 nM T50688 C7ETA1 23297736 Ki = 2 nM T50688 C0Y4GH 23297800 Ki = 650 nM T50688 CK21RA 23377844 IC50 = 210 nM T50688 CQ6M4A 23377846 IC50 = 9 nM T50688 C4OH9D 23377874 IC50 = 90 nM T50688 CMET78 23435760 IC50 = 3500 nM T50688 CKF08G 23435786 IC50 = 15000 nM T50688 CYND24 23729562 IC50 = 165 nM T50688 C96PUZ 23729563 IC50 = 30 nM T50688 CZ17YE 23731146 IC50 = 560 nM T50688 CHXT18 23731243 IC50 = 2000 nM T50688 CEA9Z8 23731244 IC50 = 12 nM T50688 CNK5O6 23731245 IC50 = 620 nM T50688 C6W9OS 23731246 IC50 = 15 nM T50688 CK7OW6 24779699 Ki = 47 nM T50688 C9L0QD 24864721 IC50 > 10000 nM T50688 CY6WR2 24872066 IC50 = 40200 nM T50688 CUM4E3 24872070 IC50 = 71700 nM T50688 CG09DH 24872646 IC50 = 77700 nM T50688 CRS65Q 24873110 IC50 = 87200 nM T50688 C0HZ7E 24873345 IC50 = 105000 nM T50688 CIS68P 25032865 IC50 > 10000 nM T50688 C07BZQ 25107507 IC50 = 2440 nM T50688 CK3FM6 25107508 IC50 = 12080 nM T50688 CN3I9J 25107569 IC50 = 15200 nM T50688 CB6H7T 25107570 IC50 = 1450 nM T50688 CC40FO 25107571 IC50 = 2000 nM T50688 C1QC4Y 25107572 IC50 = 1200 nM T50688 CKJ04T 25107573 IC50 > 100000 nM T50688 CN8Y0B 25107634 IC50 = 1780 nM T50688 C84XCZ 25107635 IC50 = 39000 nM T50688 CCY26A 25107636 IC50 > 100000 nM T50688 CO03GM 25107637 IC50 = 36500 nM T50688 CNR43C 25107638 IC50 = 2850 nM T50688 CDAC04 25107705 IC50 = 1690 nM T50688 CYS45L 25107706 IC50 = 28400 nM T50688 CYS98D 25107707 IC50 > 100000 nM T50688 CRV78W 25107708 IC50 = 54000 nM T50688 CF85WU 25107709 IC50 = 29300 nM T50688 C23YAU 25107770 IC50 = 11300 nM T50688 CQZ70E 25107771 IC50 = 9110 nM T50688 CEK7G5 25107772 IC50 = 14000 nM T50688 C3V7JU 25107773 IC50 = 2800 nM T50688 CM37RS 42607047 IC50 = 6100 nM T50688 C7K4HE 42607050 IC50 = 13000 nM T50688 CU12VE 44265226 IC50 = 0.89 nM T50688 C2POH5 44265246 IC50 = 4.76 nM T50688 CGXU38 44265249 IC50 = 0.55 nM T50688 C2E7AU 44265252 IC50 = 1 nM T50688 CD42GT 44265261 IC50 = 0.12 nM T50688 CW7O2R 44265293 IC50 = 0.57 nM T50688 CD0H6O 44268215 IC50 = 28900 nM T50688 CJ61GR 44268230 IC50 = 238 nM T50688 CRM0K3 44268269 IC50 = 25 nM T50688 C8TF4A 44268270 IC50 = 11900 nM T50688 CXP9A4 44268271 IC50 = 25 nM T50688 CVFP98 44268272 IC50 = 4 nM T50688 C5EM9S 44268276 IC50 = 252 nM T50688 CC7DE0 44268284 IC50 = 25 nM T50688 C5BM8E 44268287 IC50 > 50000 nM T50688 CJ6Z2H 44268288 IC50 > 50000 nM T50688 C2IVR7 44268289 IC50 = 17 nM T50688 CA4YL6 44268290 IC50 = 1200 nM T50688 C1LVS0 44268294 IC50 = 106 nM T50688 CP5X7D 44268296 IC50 = 225 nM T50688 CEZ7N8 44268297 IC50 = 47 nM T50688 C73WBY 44268298 IC50 = 1800 nM T50688 CS2ZJ9 44268312 IC50 = 17 nM T50688 CLJ7Y2 44268313 IC50 = 90 nM T50688 CCAR38 44268323 IC50 = 87 nM T50688 C6WRH9 44268328 IC50 = 1500 nM T50688 CH37FJ 44268364 IC50 = 4200 nM T50688 CK5IS7 44268370 IC50 = 136 nM T50688 CTD26Z 44268372 IC50 = 254 nM T50688 CRE92V 44268373 IC50 = 873 nM T50688 CC5LU4 44268375 IC50 = 320 nM T50688 CH75WX 44268376 IC50 = 447 nM T50688 CKY45X 44274285 IC50 = 3 nM T50688 CT6BV5 44279130 IC50 > 25000 nM T50688 CJY68U 44279133 IC50 = 40 nM T50688 CUB27L 44279166 IC50 = 130 nM T50688 CZ0FM9 44279167 IC50 = 3000 nM T50688 CWY2K6 44279184 IC50 > 25000 nM T50688 C7ES8I 44279259 IC50 = 70 nM T50688 C7B6NR 44279334 IC50 = 30 nM T50688 CT9RZ4 44279442 IC50 = 40 nM T50688 C42DBS 44279484 IC50 = 20 nM T50688 CC8PD2 44279492 IC50 = 6700 nM T50688 C54NRA 44279715 IC50 = 950 nM T50688 C1UJ3V 44279716 IC50 > 25000 nM T50688 CG0DB7 44279740 IC50 = 30 nM T50688 CSX2U6 44279775 IC50 = 8400 nM T50688 C2D3ML 44280044 IC50 = 250 nM T50688 C9XS5E 44281584 IC50 = 229.09 nM T50688 C31-JUL 44281660 IC50 = 270 nM T50688 C9GC6L 44281698 IC50 = 120 nM T50688 C90AZN 44281715 IC50 = 158.49 nM T50688 C7LP6X 44281716 IC50 = 640 nM T50688 CZ03QI 44281717 IC50 = 4500 nM T50688 C1MIW6 44282009 IC50 = 75.86 nM T50688 CX2PV9 44282032 IC50 = 130 nM T50688 C48KBZ 44283063 IC50 = 9.6 nM T50688 CF7C8I 44283067 IC50 = 15.6 nM T50688 C2FV0E 44283118 IC50 = 25000 nM T50688 CK0RD4 44283161 IC50 = 38 nM T50688 CXE01A 44283190 IC50 = 15.1 nM T50688 C12RPS 44283197 IC50 = 233 nM T50688 C4VW3I 44283198 IC50 = 181 nM T50688 C9ZQW4 44283202 IC50 = 11 nM T50688 C6KLR5 44283203 IC50 = 7 nM T50688 CMV19L 44283204 IC50 = 45 nM T50688 CNI3F9 44283232 IC50 = 80 nM T50688 C74CWT 44283235 IC50 = 0.71 nM T50688 CN45TM 44283254 IC50 = 69 nM T50688 CVS5P4 44283263 IC50 = 641 nM T50688 CX2PH8 44283275 IC50 = 121 nM T50688 CH29QO 44283299 IC50 = 152 nM T50688 C7FCI9 44283300 IC50 = 9.1 nM T50688 C2M4JN 44283364 IC50 = 528 nM T50688 C5R6PO 44283380 IC50 = 125 nM T50688 C09EHM 44283639 IC50 = 661 nM T50688 C20PIF 44285420 IC50 = 1000 nM T50688 C6MH2U 44285421 IC50 = 15848.93 nM T50688 CA3TB7 44285426 IC50 = 39810.72 nM T50688 CNQ7E3 44285443 IC50 = 2511.89 nM T50688 C5EG0I 44285469 IC50 < 10000 nM T50688 CC2WX5 44285470 IC50 = 25.12 nM T50688 CAD27K 44285483 IC50 = 1584.89 nM T50688 CWD58N 44285484 IC50 = 1995.26 nM T50688 CF3W1R 44285487 IC50 = 199.53 nM T50688 C4CYX6 44285495 IC50 = 1000 nM T50688 C46ICR 44285506 IC50 = 1258.93 nM T50688 CAE80Z 44285637 IC50 = 250 nM T50688 CH53NW 44285682 IC50 = 3981.07 nM T50688 C8ABI1 44287422 IC50 = 20000 nM T50688 CYAQ68 44287423 IC50 = 29900 nM T50688 C3X2LJ 44287428 IC50 = 50000 nM T50688 CQ3AF6 44287550 IC50 = 24000 nM T50688 C5PCQ0 44287569 IC50 = 8 nM T50688 C29LXN 44287570 IC50 = 28 nM T50688 CQL21H 44287634 IC50 = 20000 nM T50688 C7YE0G 44287879 IC50 = 2700 nM T50688 CTQV91 44290954 IC50 = 1220 nM T50688 CE3K5Y 44290956 IC50 > 100000 nM T50688 CNFY65 44291131 IC50 = 5000 nM T50688 CY98UX 44291379 IC50 = 120 nM T50688 CE3FQ7 44291381 IC50 = 510 nM T50688 C7XC0O 44291383 IC50 = 560 nM T50688 C6D0JM 44291385 IC50 = 1070 nM T50688 CK26HJ 44291464 IC50 > 100000 nM T50688 CKO25V 44291466 IC50 = 2 nM T50688 CM7H6A 44291467 IC50 > 100000 nM T50688 C9ZF8D 44291479 IC50 = 5 nM T50688 C7FIO4 44291481 IC50 = 20 nM T50688 C39PZH 44291483 IC50 = 40 nM T50688 C6O9CT 44291485 IC50 = 20 nM T50688 CUZ73G 44291499 IC50 = 2000 nM T50688 CAP83N 44291732 IC50 = 270 nM T50688 C0Q8WF 44291756 IC50 = 110 nM T50688 C6PHG5 44291757 IC50 = 78000 nM T50688 CQ2XC4 44291759 IC50 = 770 nM T50688 C5SM4O 44294710 IC50 = 96 nM T50688 C1CO9H 44294758 IC50 = 120 nM T50688 C6Y9PG 44294759 IC50 = 70 nM T50688 CO0JI2 44294760 IC50 = 3000 nM T50688 C37PMJ 44295006 IC50 = 200 nM T50688 CJ4PE2 44295049 IC50 = 25000 nM T50688 CR7QI4 44295086 IC50 > 20000 nM T50688 CVE2D8 44295087 IC50 = 1600 nM T50688 CHB3R8 44295112 IC50 = 470 nM T50688 C8N3TI 44295122 IC50 = 3 nM T50688 CZA76L 44295135 IC50 > 20000 nM T50688 CYF93D 44295211 IC50 > 25000 nM T50688 C8N3ZC 44295212 IC50 = 2000 nM T50688 C89PDG 44295213 IC50 = 3000 nM T50688 CTN25K 44295235 IC50 = 220 nM T50688 CD91SB 44296029 Ki = 11000 nM T50688 CESC21 44296030 Ki = 1100 nM T50688 C0NBT5 44296032 Ki = 8200 nM T50688 C0EIC6 44296106 Ki = 160000 nM T50688 CDX37F 44296107 Ki = 8500 nM T50688 CXM37J 44296126 Ki = 14000 nM T50688 CBY2N4 44296179 Ki = 5000 nM T50688 C1BDP7 44296242 Ki = 41500 nM T50688 C0R6QX 44296243 Ki = 32000 nM T50688 CYA4E9 44296248 Ki = 8000 nM T50688 CAFV23 44296408 IC50 > 3000 nM T50688 C74ZEK 44296431 IC50 > 3000 nM T50688 CFN8Q6 44296449 Ki = 3650 nM T50688 C1YD3S 44296450 Ki > 50000 nM T50688 CYSG84 44296458 IC50 > 3000 nM T50688 C4FI2N 44296514 IC50 > 3000 nM T50688 C9U3QW 44296519 IC50 > 3000 nM T50688 CQHJ16 44296532 IC50 > 3000 nM T50688 CX0Q1T 44296543 Ki = 40500 nM T50688 C2TE9R 44296548 IC50 > 3000 nM T50688 C5GY7H 44296579 IC50 > 3000 nM T50688 CYZT93 44296580 IC50 > 3000 nM T50688 C7S1JY 44296604 IC50 > 3000 nM T50688 CP89DV 44296642 IC50 > 3000 nM T50688 C1KYA3 44296682 IC50 = 10000 nM T50688 CH0JP8 44296684 IC50 = 180 nM T50688 CC0TN6 44296689 IC50 = 10000 nM T50688 CUEC26 44296697 IC50 = 350 nM T50688 C2NU5B 44296726 IC50 = 550 nM T50688 CZ17IX 44296740 IC50 > 3000 nM T50688 C3A7PY 44296742 IC50 = 10000 nM T50688 CAH14O 44296744 IC50 = 850 nM T50688 CZG93V 44296762 IC50 > 10000 nM T50688 CJRK46 44296797 IC50 > 10000 nM T50688 CY26ES 44296824 IC50 > 3000 nM T50688 CCEF03 44296851 IC50 > 3000 nM T50688 C27UPR 44296852 IC50 > 3000 nM T50688 C0FK5Q 44296857 IC50 > 3000 nM T50688 CR9U6E 44296858 IC50 > 3000 nM T50688 CS2E4W 44296864 IC50 > 10000 nM T50688 CS62KL 44296866 IC50 = 5000 nM T50688 C0KY3B 44296868 IC50 > 10000 nM T50688 C27HKT 44296892 IC50 = 200 nM T50688 CVAF21 44296901 IC50 > 3000 nM T50688 C5O8IC 44296903 IC50 > 3000 nM T50688 C4ZG0D 44297806 IC50 = 1100 nM T50688 CC4LU8 44297807 IC50 = 1600 nM T50688 C6F1CD 44297814 IC50 = 10000 nM T50688 CGZ82H 44297845 IC50 = 300000 nM T50688 C0KX7H 44297846 IC50 = 530 nM T50688 CY35IN 44297847 IC50 = 2000 nM T50688 CX2PK9 44300973 IC50 = 7000 nM T50688 CA78QS 44300974 IC50 > 10000 nM T50688 CPJU95 44300981 IC50 > 10000 nM T50688 C9YT1L 44300986 IC50 = 65 nM T50688 CWP15R 44301007 IC50 = 19 nM T50688 CL84GY 44301008 IC50 = 28 nM T50688 CSCA61 44301010 IC50 > 10000 nM T50688 CX3Y4B 44301021 IC50 = 27 nM T50688 CPW8S2 44301026 IC50 = 9 nM T50688 CP1F5U 44301032 IC50 = 57 nM T50688 COX26S 44301040 IC50 = 15 nM T50688 C9OU5P 44301044 IC50 = 12 nM T50688 CO6HW2 44301065 Ki = 2.3 nM T50688 CWP52F 44301068 IC50 = 9000 nM T50688 CLCO73 44301083 IC50 > 10000 nM T50688 C6DZ3F 44301106 IC50 = 11 nM T50688 CC4LO8 44301244 IC50 = 3000 nM T50688 CIJ28H 44301270 IC50 = 13 nM T50688 C4W3LK 44301283 IC50 = 51 nM T50688 C7VC5T 44301286 IC50 > 10000 nM T50688 CBT2O3 44301295 IC50 = 15 nM T50688 CI39XL 44301310 IC50 > 10000 nM T50688 CZ14EM 44301350 IC50 > 10000 nM T50688 C3MSY1 44301352 IC50 = 8 nM T50688 C5OA0I 44301363 IC50 = 81 nM T50688 C0G3LI 44301379 IC50 = 8 nM T50688 CWBC76 44301520 Ki = 2.1 nM T50688 C9QIP0 44303539 IC50 = 500 nM T50688 CC3H4P 44303550 IC50 = 105 nM T50688 C39FGB 44303551 IC50 = 1350 nM T50688 CA3X5V 44303563 IC50 = 40 nM T50688 C4AO7I 44303592 IC50 = 17 nM T50688 CPX4L1 44303611 IC50 = 65 nM T50688 CRJP53 44303836 IC50 = 17 nM T50688 CTBK03 44303837 IC50 = 35 nM T50688 CO5KC2 44304468 IC50 = 20000 nM T50688 CR30VX 44304469 IC50 = 6 nM T50688 CC9H7K 44304480 IC50 = 3.5 nM T50688 CJ68BM 44304481 IC50 = 0.5 nM T50688 CYKT90 44304483 IC50 = 4.7 nM T50688 CA09ZS 44304485 IC50 = 210 nM T50688 C5TY8F 44304495 IC50 = 434 nM T50688 CK7YC1 44304496 IC50 = 12 nM T50688 C4E1TI 44304497 IC50 = 18 nM T50688 CEY8V5 44304498 IC50 = 1.4 nM T50688 CT5KO2 44304499 IC50 = 500 nM T50688 CPD08J 44304500 IC50 = 25 nM T50688 CE42YV 44304526 IC50 = 35 nM T50688 CB3A9F 44304531 IC50 = 6 nM T50688 CBZ12F 44304532 IC50 = 11.4 nM T50688 C3FJ5K 44304541 IC50 = 80 nM T50688 CEX49N 44304547 IC50 = 75000 nM T50688 CSNM29 44304548 IC50 = 14 nM T50688 C5KQ1N 44304549 IC50 = 4850 nM T50688 C1IYO2 44304571 IC50 = 5.7 nM T50688 CZG56O 44304572 IC50 = 260 nM T50688 CR25CI 44304573 IC50 = 4600 nM T50688 C8KS3L 44304576 IC50 = 75 nM T50688 C1K4WA 44304587 IC50 = 20 nM T50688 C12GLJ 44304588 IC50 = 7.5 nM T50688 C0WA7Z 44304604 IC50 = 110 nM T50688 C47YWJ 44304607 IC50 = 31 nM T50688 CFPV93 44304608 IC50 = 5.6 nM T50688 CE1N6V 44304609 IC50 = 43 nM T50688 C21SEM 44304613 IC50 = 5.3 nM T50688 CFC0P2 44304619 IC50 = 12 nM T50688 C2G4XE 44304624 IC50 = 6.6 nM T50688 CM78IK 44304645 IC50 = 33 nM T50688 CR9Z7P 44304646 IC50 = 100 nM T50688 CF82AW 44304647 IC50 = 2.9 nM T50688 CGRU80 44304650 IC50 = 2.6 nM T50688 CY2R9X 44304655 IC50 = 70 nM T50688 CC5B3K 44304656 IC50 = 150 nM T50688 CFTN27 44304659 IC50 = 4780 nM T50688 CL5K9N 44304660 IC50 = 4 nM T50688 C3E5VJ 44304661 IC50 = 22 nM T50688 CAVK91 44304674 IC50 = 38 nM T50688 CTY01P 44304675 IC50 = 6.8 nM T50688 CWCM82 44304679 IC50 = 4 nM T50688 CKR7Y0 44304718 IC50 = 1.6 nM T50688 CS30ZM 44304723 IC50 = 3 nM T50688 CLI42H 44304724 IC50 = 35 nM T50688 C8A3KN 44304725 IC50 = 310 nM T50688 CX1E3B 44304726 IC50 = 9.5 nM T50688 CKN1E4 44304733 IC50 = 590 nM T50688 CE87NH 44304744 IC50 = 19 nM T50688 C7FOJ3 44304745 IC50 = 132 nM T50688 C1VY6U 44304785 IC50 = 4.5 nM T50688 CPS9C0 44304808 IC50 = 5.4 nM T50688 C1NFJ0 44304842 IC50 = 4 nM T50688 CMZC63 44304843 IC50 = 2.8 nM T50688 CK68QA 44304844 IC50 = 2.7 nM T50688 CRN6V1 44304845 IC50 = 7 nM T50688 C5YNE8 44304874 IC50 = 1 nM T50688 CEA9H3 44304875 IC50 = 29 nM T50688 CMTQ46 44304901 IC50 = 8 nM T50688 C2H8DU 44304902 IC50 = 28 nM T50688 C0CMR7 44304903 IC50 = 1060 nM T50688 CX69MO 44304904 IC50 = 22 nM T50688 CVDR16 44304905 IC50 = 3.6 nM T50688 C8RYE9 44304952 IC50 = 17 nM T50688 CG2N3X 44304953 IC50 = 500 nM T50688 CME60P 44304954 IC50 = 231 nM T50688 CS12DA 44305003 IC50 = 2.5 nM T50688 CM67BS 44305004 IC50 = 12 nM T50688 CH0F7S 44305008 IC50 = 103 nM T50688 CF9ZI0 44305062 IC50 = 4185 nM T50688 CG6P3Y 44305143 IC50 = 4 nM T50688 CI3OA0 44305239 IC50 = 1700 nM T50688 CIF0U5 44305476 IC50 = 49 nM T50688 CWF31T 44305508 IC50 = 140 nM T50688 C5Y3IP 44305645 IC50 = 2700 nM T50688 CP5O4B 44305658 IC50 = 3300 nM T50688 CQOS32 44305694 IC50 = 31 nM T50688 C1A5QE 44305716 IC50 = 44 nM T50688 CA82VR 44305726 IC50 = 210 nM T50688 CB21HD 44305872 IC50 = 35000 nM T50688 CJ9C1D 44306030 IC50 = 7000 nM T50688 CM9ZV1 44306543 IC50 = 707945.78 nM T50688 CX40ZQ 44306545 IC50 = 30199.52 nM T50688 CO8LM1 44306547 IC50 = 741310.24 nM T50688 C5QM2G 44306568 IC50 = 100 nM T50688 CUY0W7 44306569 IC50 = 200 nM T50688 CL59SB 44306616 IC50 = 758577.58 nM T50688 C6K3TO 44306710 IC50 = 7585.78 nM T50688 CP09ST 44306715 IC50 = 52480.75 nM T50688 CCH6E0 44306731 IC50 = 100 nM T50688 CE78JY 44306747 IC50 = 100000 nM T50688 CD6C2J 44306765 IC50 = 200 nM T50688 C9F5ZP 44306766 IC50 = 2000 nM T50688 CCU8M2 44306772 IC50 = 630.96 nM T50688 CC9N4L 44306786 IC50 = 302 nM T50688 C0BXH2 44306842 IC50 = 363.08 nM T50688 CL3AD9 44306932 IC50 = 128.82 nM T50688 C19BET 44306947 IC50 = 199526.23 nM T50688 CLM91S 44307016 IC50 = 1905.46 nM T50688 C7L5JI 44307035 IC50 = 9120.11 nM T50688 CAD8H2 44307043 IC50 = 6456.54 nM T50688 CHLY12 44307056 IC50 = 5011.87 nM T50688 C8WD1N 44307070 IC50 = 5248.07 nM T50688 C3YZB0 44307099 IC50 = 91201.08 nM T50688 CBZ6D8 44307217 IC50 = 3467.37 nM T50688 CIX09R 44307237 IC50 = 2511.89 nM T50688 CN36PV 44307238 IC50 = 239.88 nM T50688 C0DGS2 44307241 IC50 = 794.33 nM T50688 CJ7BQ2 44307259 IC50 = 109647.82 nM T50688 C8A5MJ 44307296 IC50 = 758577.58 nM T50688 C80FZA 44307297 IC50 = 33113.11 nM T50688 CI59NO 44307365 IC50 = 4073.8 nM T50688 C6B5JQ 44315195 IC50 = 2.7 nM T50688 CK2B7R 44315447 IC50 = 2.6 nM T50688 CMZJ69 44315702 IC50 = 23.7 nM T50688 CJN6H3 44315779 IC50 = 2 nM T50688 C8LQ3E 44315780 IC50 = 20 nM T50688 C5XE1O 44315792 IC50 = 20 nM T50688 CPT6R4 44315793 IC50 = 20 nM T50688 C2TE0B 44316045 IC50 = 6 nM T50688 C7P1CL 44316059 IC50 = 7 nM T50688 CDVZ48 44316106 IC50 = 2 nM T50688 C9B8CD 44316156 IC50 = 5 nM T50688 CUBM67 44316184 IC50 = 3 nM T50688 CA0P1Z 44316450 IC50 = 52 nM T50688 CAI6P7 44316522 IC50 = 4.8 nM T50688 C8DRY2 44316532 IC50 = 4 nM T50688 CYTL98 44316560 IC50 = 200 nM T50688 C6QU9I 44316563 IC50 > 50000 nM T50688 C4U2XO 44316579 IC50 = 224 nM T50688 C13IEA 44317739 IC50 = 8 nM T50688 C5UTI9 44318089 IC50 = 16 nM T50688 C9XH0Y 44318100 IC50 = 32 nM T50688 CZ5R4V 44318107 IC50 = 129 nM T50688 C97YTO 44318110 IC50 = 53 nM T50688 COB28I 44318124 IC50 = 47 nM T50688 CA65ZG 44318139 IC50 = 78 nM T50688 CMO5P7 44318169 IC50 = 630 nM T50688 CR3D0I 44319347 IC50 = 41 nM T50688 CT73SX 44319352 IC50 = 260 nM T50688 CAP0X7 44319363 IC50 = 56 nM T50688 C20MFD 44319365 IC50 = 1700 nM T50688 CJUP56 44319437 IC50 = 680 nM T50688 CV9CP5 44319448 IC50 = 100 nM T50688 C58SYJ 44319608 IC50 = 1800 nM T50688 CFN08C 44319632 IC50 = 220 nM T50688 CS67MW 44320027 IC50 > 1000 nM T50688 C91SAN 44320056 IC50 > 1000 nM T50688 CC4UG8 44320077 IC50 > 1000 nM T50688 CAVD13 44320155 IC50 > 1000 nM T50688 C95KAZ 44320173 IC50 = 88 nM T50688 CSV1C2 44320174 IC50 > 1000 nM T50688 C7GXI5 44320211 IC50 = 540 nM T50688 CWS24X 44320274 IC50 > 1000 nM T50688 C1W8ID 44320282 IC50 = 30 nM T50688 C6F7OI 44320305 IC50 = 340 nM T50688 CN08CV 44320306 IC50 > 1000 nM T50688 CVX0F7 44320364 IC50 = 720 nM T50688 C3SXG5 44320893 IC50 = 18 nM T50688 C5FAY7 44321219 IC50 > 1000 nM T50688 CC25UD 44321220 IC50 > 1000 nM T50688 C8X5IP 44321235 IC50 > 100 nM T50688 CME9U8 44321274 IC50 = 6 nM T50688 C82THY 44321295 IC50 = 8.7 nM T50688 CN41VK 44321296 IC50 = 1.4 nM T50688 CA5ZE4 44321313 IC50 = 62 nM T50688 CSX9Z2 44321328 IC50 = 9.8 nM T50688 CM8P0R 44321368 IC50 = 100 nM T50688 C5PBW9 44321507 IC50 > 100 nM T50688 C26IPS 44321551 IC50 > 100 nM T50688 C5ZAL0 44321567 IC50 = 730 nM T50688 C7UOZ5 44321682 IC50 > 100 nM T50688 C4BTK5 44321683 IC50 = 42 nM T50688 CFSI83 44321913 IC50 = 440 nM T50688 CIX50Z 44321934 IC50 = 2.7 nM T50688 C82IOL 44322337 IC50 = 0.6 nM T50688 C7PYO4 44322627 IC50 = 0.12 nM T50688 C5AG3Y 44322644 IC50 = 0.51 nM T50688 CKY2F1 44329896 Ki > 25000 nM T50688 CKXQ61 44329897 Ki > 25000 nM T50688 C79CIF 44329957 IC50 > 10000 nM T50688 C91OLV 44329959 IC50 > 10000 nM T50688 CUQ2M9 44330009 IC50 = 7100 nM T50688 CUK74V 44330015 Ki = 2100 nM T50688 C38PGY 44330039 Ki > 25000 nM T50688 CF9SY3 44330086 Ki > 25000 nM T50688 CAT6Y2 44330200 Ki > 25000 nM T50688 CSIG14 44333548 IC50 > 10000 nM T50688 C2E3VH 44333550 IC50 = 1700 nM T50688 C23DVQ 44333621 IC50 > 10000 nM T50688 C4X3KB 44333751 IC50 = 860 nM T50688 CY84IA 44333752 IC50 > 10000 nM T50688 CLE04Q 44333753 IC50 = 5200 nM T50688 CE8G2W 44336187 IC50 = 68200 nM T50688 C67WVQ 44336210 IC50 > 200000 nM T50688 CUG16W 44336218 Ki = 780 nM T50688 C3V7ZN 44336250 IC50 > 200000 nM T50688 C9KXF4 44336279 IC50 = 52000 nM T50688 C7D6EU 44336336 Ki = 5300 nM T50688 CHDR52 44336478 IC50 > 10000 nM T50688 CB5QP3 44336511 IC50 > 10000 nM T50688 C2R8GS 44336762 IC50 > 10000 nM T50688 CW9RO6 44336769 IC50 = 90 nM T50688 C52LJU 44336770 IC50 > 8000 nM T50688 CDLE79 44337733 Ki = 47000 nM T50688 CN0K7Q 44337734 Ki = 30000 nM T50688 CY5R8E 44337742 Ki = 29000 nM T50688 CAQZ60 44337758 Ki = 2750 nM T50688 CA47BJ 44337773 Ki = 28000 nM T50688 C4LEU0 44340569 IC50 = 667 nM T50688 CTRQ17 44341096 IC50 = 198000 nM T50688 CX46NY 44343237 IC50 > 25000 nM T50688 CPW4H8 44343633 IC50 = 59 nM T50688 C0R2ZS 44343700 IC50 = 20 nM T50688 CO8P3W 44343737 IC50 = 3.5 nM T50688 CG83NM 44343750 IC50 = 50 nM T50688 C6IC2T 44343773 IC50 = 160 nM T50688 C95EFU 44343896 IC50 > 90 nM T50688 CELV48 44350342 IC50 > 1000000 nM T50688 CP4R1A 44350344 IC50 = 1400 nM T50688 CDE56C 44350392 IC50 = 34000 nM T50688 CEP6G1 44350415 IC50 > 100000 nM T50688 C7J9NH 44350447 IC50 = 7300 nM T50688 CH6UX8 44350448 IC50 = 11000 nM T50688 C4C2PF 44350449 IC50 = 5600 nM T50688 CP4TD3 44350450 IC50 > 100000 nM T50688 C2V8FY 44350717 IC50 = 330 nM T50688 CMLD50 44350731 IC50 = 1200 nM T50688 CEFL68 44351621 IC50 > 200000 nM T50688 CCQ08X 44351628 Ki = 4 nM T50688 CH1O6S 44351664 Ki = 1900 nM T50688 C61BOQ 44351682 Ki = 106 nM T50688 C6SN9U 44351704 Ki = 271 nM T50688 CM5X6P 44351788 IC50 = 76600 nM T50688 C8XB4U 44351866 Ki = 3130 nM T50688 C1QGR5 44351885 IC50 = 17700 nM T50688 C9FUW5 44352004 IC50 = 70000 nM T50688 CEQ93X 44353584 IC50 = 2400 nM T50688 CCAZ98 44359505 IC50 = 1100 nM T50688 CTI3C9 44359535 IC50 = 5200 nM T50688 CK04UD 44359546 IC50 = 39000 nM T50688 CB42IU 44359616 IC50 = 6400 nM T50688 CA1DP5 44359630 IC50 = 2500 nM T50688 CZ68AH 44359656 IC50 = 3700 nM T50688 CIPX97 44359766 IC50 > 100000 nM T50688 CNLV75 44359767 IC50 > 100000 nM T50688 CV8JY9 44362649 IC50 = 1300 nM T50688 C68QVP 44362650 IC50 = 15000 nM T50688 CPT04Y 44362651 IC50 = 45000 nM T50688 C35BCT 44362902 IC50 = 14000 nM T50688 C3TSZ6 44362908 IC50 = 170 nM T50688 CTO32M 44362922 IC50 = 510 nM T50688 C80OTL 44362923 IC50 = 170 nM T50688 CI2UG4 44362951 IC50 > 300000 nM T50688 CY07RK 44363126 Ki = 8 nM T50688 CN9M2P 44363186 Ki = 90 nM T50688 CIY64N 44364493 IC50 = 110 nM T50688 CSRM97 44364562 IC50 = 140 nM T50688 C6EUK9 44364573 IC50 = 229.09 nM T50688 CXO4Y9 44364601 IC50 = 4466.84 nM T50688 C1LIW7 44364621 IC50 = 63 nM T50688 C6IFM5 44364673 IC50 = 6.1 nM T50688 C92MKD 44364694 IC50 = 210 nM T50688 CI7BH0 44364738 IC50 = 1500 nM T50688 CHK71U 44365992 IC50 = 17.9 nM T50688 C3E1ID 44366016 IC50 = 0.37 nM T50688 CT7DQ8 44366048 IC50 = 48 nM T50688 C2QNL7 44366077 IC50 = 0.36 nM T50688 CU0WI3 44366139 IC50 = 66.8 nM T50688 CD8RZ0 44366167 IC50 = 0.24 nM T50688 C1WHZ3 44366226 IC50 = 13.5 nM T50688 C3AM0D 44366227 IC50 = 0.1 nM T50688 CZH23I 44366235 IC50 = 0.1 nM T50688 CT58MH 44366375 IC50 = 0.5 nM T50688 CNZQ89 44366409 IC50 = 157 nM T50688 C1J2CW 44366410 IC50 > 10000 nM T50688 CN2L3U 44367917 Ki = 500 nM T50688 CVGB31 44368140 Ki = 2 nM T50688 CO1SR9 44368152 Ki > 50000 nM T50688 CB0TF6 44368570 IC50 = 776 nM T50688 C47OWF 44368757 IC50 > 10000 nM T50688 CAS01N 44372658 IC50 = 21000 nM T50688 CGIP26 44372909 IC50 = 10400 nM T50688 CYD6H2 44372941 IC50 = 30000 nM T50688 C4NU0I 44372954 IC50 = 81000 nM T50688 C6B5FO 44372955 IC50 = 31000 nM T50688 CFO34W 44372962 IC50 = 100000 nM T50688 COYQ79 44372977 IC50 = 30000 nM T50688 CHS2V0 44373024 IC50 > 30000 nM T50688 C8WQ3F 44373152 IC50 = 8900 nM T50688 CKR0X7 44373170 IC50 = 87000 nM T50688 C6X9UK 44373176 IC50 = 24000 nM T50688 CAIJ06 44373182 IC50 > 30000 nM T50688 C09MLI 44373256 IC50 = 30000 nM T50688 C89GTD 44373300 IC50 > 100000 nM T50688 CU12HA 44373303 IC50 = 19000 nM T50688 C68DAQ 44373341 IC50 = 45000 nM T50688 CQE4R3 44373603 IC50 = 30000 nM T50688 C4V3KU 44373605 IC50 = 30000 nM T50688 CJC35L 44376533 IC50 = 0.54 nM T50688 CXON13 44376539 IC50 = 0.36 nM T50688 C4D2SH 44376550 IC50 = 1 nM T50688 C68SYL 44376551 IC50 = 0.36 nM T50688 CJA9Q6 44376578 IC50 = 7.6 nM T50688 CA3UC1 44376579 IC50 = 1.7 nM T50688 CHV7T9 44376681 IC50 = 2.2 nM T50688 CA5FS3 44376772 IC50 = 48000 nM T50688 CC0WL9 44376773 IC50 = 0.37 nM T50688 CHZ0Q1 44376790 IC50 = 7.9 nM T50688 C8O7TA 44378089 Ki = 110 nM T50688 C7HTK1 44378106 Ki = 2650 nM T50688 C5XJ1T 44378195 Ki = 2.1 nM T50688 C7L5ZE 44378218 Ki = 26 nM T50688 C8MJ9S 44378222 Ki = 65 nM T50688 CJE6O9 44378223 Ki = 25300 nM T50688 CWK48R 44378224 Ki = 820 nM T50688 C4PIV6 44378302 Ki > 10000 nM T50688 C2X4KT 44378303 Ki = 82 nM T50688 CAE13J 44378307 Ki = 27 nM T50688 CQ3EA4 44378320 Ki = 9.5 nM T50688 CPAQ56 44378327 Ki = 15100 nM T50688 CM5YQ1 44378331 Ki = 2.5 nM T50688 CD6C9K 44378336 Ki = 7040 nM T50688 C7CTJ8 44378360 Ki > 100000 nM T50688 C4K6LW 44378361 Ki = 280 nM T50688 CTZO38 44378378 Ki = 1250 nM T50688 C89JAB 44378400 Ki = 430 nM T50688 C7O9AP 44378401 Ki = 20 nM T50688 C3C8VJ 44378494 Ki = 188 nM T50688 C4SKJ9 44378558 Ki = 2.1 nM T50688 CL9UT4 44378583 Ki = 135 nM T50688 C42USR 44378584 Ki = 77 nM T50688 CN9Z4W 44378585 Ki = 610 nM T50688 CR51ID 44378699 IC50 = 16 nM T50688 CAO29R 44378701 IC50 = 150 nM T50688 CWP41H 44378720 IC50 = 3 nM T50688 C2U6ZA 44378747 IC50 = 14 nM T50688 CT9H2B 44378748 IC50 = 3 nM T50688 CNS75M 44378858 IC50 = 20 nM T50688 CENU52 44378961 IC50 = 2 nM T50688 C3UQT1 44378995 IC50 = 38 nM T50688 CHC7N5 44379066 IC50 = 430 nM T50688 CSA20X 44381676 IC50 = 109.65 nM T50688 CZTW31 44381688 IC50 = 39.81 nM T50688 C6R8KC 44381737 IC50 = 85.11 nM T50688 CY1U0D 44381774 IC50 = 114.82 nM T50688 CL9FU3 44381783 IC50 = 40.74 nM T50688 CMB53C 44381797 IC50 = 38.02 nM T50688 CQ9UO5 44381825 IC50 = 151.36 nM T50688 CQ06HD 44381864 IC50 = 125.89 nM T50688 C42PBL 44381878 IC50 = 331.13 nM T50688 CKE79T 44381879 IC50 = 190.55 nM T50688 CS9V1U 44381881 IC50 = 380 nM T50688 CS51QV 44381885 IC50 = 18197.01 nM T50688 CLGQ87 44381898 IC50 = 29000 nM T50688 C84FJL 44381902 IC50 = 134.9 nM T50688 CJ5MH7 44381905 IC50 = 40.74 nM T50688 CDV3U9 44381908 IC50 = 130 nM T50688 CN5EU2 44381918 IC50 = 34 nM T50688 C4TCZ8 44381942 IC50 = 230000 nM T50688 C48UAI 44381947 IC50 = 75.86 nM T50688 C8B3LU 44381948 IC50 = 42.66 nM T50688 C45BHN 44381953 IC50 = 9200 nM T50688 C9ZOW8 44381959 IC50 = 40.74 nM T50688 CQ08VO 44381964 IC50 = 1659.59 nM T50688 CP3D6M 44381975 IC50 = 33113.11 nM T50688 C5ERH4 44381977 IC50 = 44.67 nM T50688 C6ECI7 44381991 IC50 = 37.15 nM T50688 C1NXQ2 44381992 IC50 = 2800 nM T50688 C6K4IV 44382000 IC50 = 186.21 nM T50688 CNQY28 44382002 IC50 = 707.95 nM T50688 C5O1SY 44382014 IC50 = 30.9 nM T50688 CN21FS 44382015 IC50 = 38.02 nM T50688 C9D6RZ 44382030 IC50 = 79.43 nM T50688 C8RYM7 44382051 IC50 = 501.19 nM T50688 COZA49 44382083 IC50 = 40.74 nM T50688 CSW25H 44382135 IC50 = 79.43 nM T50688 CW80ED 44382136 IC50 = 79.43 nM T50688 CZB83R 44382356 IC50 = 4900 nM T50688 C3L4XR 44382357 IC50 = 270 nM T50688 C1GOE5 44382394 IC50 = 23 nM T50688 CE18UX 44382445 IC50 = 13 nM T50688 CE7L0H 44382481 IC50 = 331131.12 nM T50688 C3W0TK 44382482 IC50 > 30000 nM T50688 CWDC18 44383692 IC50 > 100000 nM T50688 CAY53C 44383697 IC50 = 3600 nM T50688 CB2KW6 44383745 IC50 = 12000 nM T50688 C3Q0GH 44383752 IC50 = 800 nM T50688 CBH12Q 44383755 IC50 = 53000 nM T50688 CY70ZS 44383803 IC50 = 2600 nM T50688 CRJ1M9 44383805 IC50 = 23000 nM T50688 CCR0M8 44383848 IC50 = 17000 nM T50688 C1E0CL 44384154 IC50 = 850 nM T50688 C28CSF 44384225 IC50 = 3500 nM T50688 CG0I7U 44384233 IC50 = 170 nM T50688 CZOH46 44384400 IC50 = 55000 nM T50688 C3VKC9 44384418 IC50 = 47000 nM T50688 CWY40J 44384448 IC50 = 3600 nM T50688 CWX1O8 44384452 IC50 = 1500 nM T50688 CR51GC 44384509 IC50 = 13000 nM T50688 C2PXN3 44384519 IC50 > 100000 nM T50688 C1SKZ8 44384644 IC50 = 690 nM T50688 CBV4X3 44384707 IC50 = 1900 nM T50688 C1U0OM 44384812 IC50 = 360 nM T50688 CD95EQ 44384863 IC50 > 100000 nM T50688 CE1LV5 44385010 IC50 = 9 nM T50688 CM27CY 44385012 IC50 = 11 nM T50688 CRO89U 44385014 IC50 = 16 nM T50688 CACQ93 44385048 IC50 = 13 nM T50688 CZIJ16 44385402 IC50 = 12000 nM T50688 CVYB52 44393453 IC50 = 170 nM T50688 CAD12L 44393517 IC50 = 25 nM T50688 CS2I9D 44394317 IC50 = 13 nM T50688 CL9GN5 44394834 IC50 = 79.3 nM T50688 CIS4X5 44394933 IC50 = 15719 nM T50688 CA30XW 44394981 IC50 = 56.4 nM T50688 C4X2PI 44395065 IC50 = 2850 nM T50688 C0IN2J 44395933 IC50 = 1100 nM T50688 CL1AJ8 44395975 IC50 = 2900 nM T50688 CK4YH8 44396023 IC50 = 870 nM T50688 C3DN8C 44396062 IC50 = 4700 nM T50688 CC62KR 44400343 Ki = 5190 nM T50688 C8OA0D 44400345 Ki = 59050 nM T50688 CK5ZW7 44400347 Ki = 3940 nM T50688 CE18LD 44407524 IC50 = 423 nM T50688 CZ4O2D 44407529 IC50 = 22 nM T50688 CV36MS 44407555 IC50 = 91 nM T50688 C9XIY5 44407556 IC50 = 64 nM T50688 C1E7HF 44407560 IC50 = 17 nM T50688 CW8MQ7 44407577 IC50 = 126 nM T50688 C03KFP 44407668 IC50 = 216 nM T50688 C7CP1X 44407779 IC50 = 1217 nM T50688 C5LF3K 44412296 IC50 = 16.2 nM T50688 C87QUH 44455076 IC50 > 10000 nM T50688 C7A1WN 44458461 IC50 = 1.2 nM T50688 CX0A3S 44458463 IC50 = 1.5 nM T50688 C6L5HF 44458472 IC50 = 102 nM T50688 CB30EA 44458473 IC50 = 0.86 nM T50688 CV9OB8 44458488 IC50 = 0.55 nM T50688 C5Y4DU 44458504 IC50 = 260 nM T50688 CMR2F1 44459058 IC50 = 9700 nM T50688 C13NVH 44459345 IC50 > 100000 nM T50688 CDKG38 44459361 IC50 = 160 nM T50688 C9G5ZA 44459507 IC50 = 240 nM T50688 C70KPC 44459508 IC50 = 270 nM T50688 C9X7AN 44459610 IC50 = 332 nM T50688 C3UHE0 44459630 IC50 = 8 nM T50688 C4YO1S 44459631 IC50 = 160 nM T50688 C8V9BY 44459642 IC50 = 250 nM T50688 CM03VR 44459643 IC50 = 100000 nM T50688 CKR0S7 44459645 IC50 = 100000 nM T50688 CQRA01 44459646 IC50 = 2400 nM T50688 C2T4XF 44459647 IC50 = 3450 nM T50688 C9MTP5 44459648 IC50 = 50000 nM T50688 CQU0Y3 44459649 IC50 = 250 nM T50688 CG5T2Y 44459650 IC50 = 319 nM T50688 CX4JZ1 44459666 IC50 = 2 nM T50688 C9WBE0 44459668 IC50 = 30000 nM T50688 CGLX83 44459727 IC50 = 9700 nM T50688 COKC08 44459728 IC50 = 5000 nM T50688 C6O8ZD 44459743 IC50 = 4 nM T50688 CMU71G 44459764 IC50 = 2 nM T50688 C4HV0D 44459765 IC50 = 830 nM T50688 C0V8SK 44459766 IC50 = 60 nM T50688 CWR7Q1 44459770 IC50 = 1 nM T50688 CAXJ53 44459773 IC50 = 7 nM T50688 CVS29Q 44459774 IC50 = 616 nM T50688 CU95CL 44459843 IC50 = 23 nM T50688 CFJC10 44459851 IC50 = 43 nM T50688 CGJ3Y7 44459852 IC50 = 210 nM T50688 C56CVI 44459873 IC50 = 1160 nM T50688 C9CAP7 44459874 IC50 = 260 nM T50688 C8XH7Y 44461765 Ki = 2.5 nM T50688 C5DA7R 44461812 Ki = 1.3 nM T50688 CH2XK6 44461891 Ki = 1.5 nM T50688 C8N6XQ 44462164 IC50 = 11 nM T50688 C1HQL7 44462165 IC50 = 28 nM T50688 C9PWK3 44462196 IC50 = 32 nM T50688 C87CFQ 44462263 IC50 = 1060 nM T50688 CY4L8W 44549109 IC50 = 61 nM T50688 C4FW5Y 44549223 IC50 = 38 nM T50688 C7IXB3 44550126 IC50 = 21.3 nM T50688 CW9N7S 44550127 IC50 = 101 nM T50688 CK4UM8 44550445 IC50 = 154 nM T50688 C3QU6T 44550446 IC50 = 36 nM T50688 CS0Z3D 44550447 IC50 = 70 nM T50688 CH9M4W 44550573 IC50 = 106 nM T50688 C5V7GK 44550574 IC50 = 121 nM T50688 CB7R0U 44550575 IC50 = 27 nM T50688 CN3T7E 44550576 IC50 = 7.3 nM T50688 CO8EM6 44550577 IC50 = 140.6 nM T50688 C4XF2A 44550689 IC50 = 355 nM T50688 C4T6XP 44550690 IC50 = 38 nM T50688 CUWQ62 44550691 IC50 = 71 nM T50688 C69RIT 44550947 IC50 = 28 nM T50688 C4U9VF 44591153 IC50 > 10000 nM T50688 CER2H0 44591154 IC50 > 10000 nM T50688 C7TX9N 44591155 IC50 > 10000 nM T50688 C5VBY3 44820665 IC50 = 95 nM T50688 CKV5P7 45264021 IC50 = 32 nM T50688 C9RHC0 45483715 IC50 = 429 nM T50688 C4E8LZ 45483796 IC50 = 25 nM T50688 CU58DV 45483797 IC50 = 51 nM T50688 C18VUC 45483798 IC50 = 20 nM T50688 C89ZFA 46224777 IC50 = 34400 nM T50688 C5X1NZ 46224858 IC50 = 121000 nM T50688 CDG6B1 46224859 IC50 = 159000 nM T50688 CKM2X1 46224860 IC50 = 14800 nM T50688 CL39GY 46224861 IC50 = 76700 nM T50688 C56PVC 46226894 IC50 > 50000 nM T50688 CVXH79 46226896 IC50 = 2300 nM T50688 CBKZ57 46226897 IC50 = 8900 nM T50688 C30JXH 46226899 IC50 = 15000 nM T50688 C2WHK1 46226900 IC50 = 9700 nM T50688 C5H9YT 46226901 IC50 = 16500 nM T50688 CV8W7P 46226902 IC50 = 7700 nM T50688 C83EWD 46226903 IC50 = 5200 nM T50688 CRVU54 46226904 IC50 = 18000 nM T50688 CE85AX 46226905 IC50 = 11800 nM T50688 C0Y1TB 46232105 IC50 = 0.56 nM T50688 CP7U9T 50907449 IC50 > 10000 nM T50688 C6XNM0 53380822 IC50 > 100000 nM T50688 C1KFQ0 53380823 IC50 > 100000 nM T50688 C7JWD0 53380936 IC50 > 100000 nM T50688 C97KGD 53380937 IC50 > 100000 nM T50688 CKV6Q2 53380938 IC50 > 100000 nM T50688 C47WIH 53380939 IC50 > 100000 nM T50688 CY3RO0 53380940 IC50 > 10000 nM T50688 C3R8PW 53380941 IC50 > 100000 nM T50688 C2G6VQ 54580191 IC50 = 0.94 nM T50688 C1D8YQ 54581193 IC50 = 0.98 nM T50688 C0YTW6 54583189 IC50 = 0.4 nM T50688 CY08RT 54586079 IC50 = 0.023 nM T50688 CY7EQ4 56658817 IC50 = 6 nM T50688 C7I1EZ 56660024 IC50 = 350 nM T50688 C6OI5V 56660094 IC50 > 100000 nM T50688 CKFI81 56660095 IC50 > 100000 nM T50688 C0RFN9 56661197 IC50 = 230 nM T50688 CRT92P 56663492 IC50 = 37 nM T50688 CJR9F6 56666913 IC50 = 6.8 nM T50688 CHO1R7 56666917 IC50 = 6.5 nM T50688 CKR2H3 56666921 IC50 = 6.5 nM T50688 CETB80 56669198 IC50 = 1.7 nM T50688 CIH3K9 56670363 IC50 = 5.5 nM T50688 CF96ZL 56672656 IC50 = 18 nM T50688 CV68RB 56676028 IC50 = 11.6 nM T50688 CTXA08 56676029 IC50 = 1.3 nM T50688 CV3B1N 56676031 IC50 = 3260 nM T50688 CR3Q0L 56677204 IC50 = 270 nM T50688 C5EPH9 56677206 IC50 = 1200 nM T50688 CDP40K 56679353 IC50 = 1.8 nM T50688 CT7U8L 56683905 IC50 > 100000 nM T50688 C3CDB4 56683906 IC50 > 100000 nM T50688 CRCK01 56949775 IC50 = 22.7 nM T50688 C64ETP 56949776 EC50 = 40.8 nM T50688 CI2Z8J 56949777 IC50 = 62.5 nM T50688 C6A8YO 56949924 IC50 = 136 nM T50688 CPBN64 56949925 IC50 = 1154 nM T50688 C54RZY 56949926 IC50 = 1322 nM T50688 CM90UN 57390370 IC50 = 1.2 nM T50688 CB57DW 57391171 IC50 = 1500 nM T50688 CWJ4I7 57391565 IC50 = 3400 nM T50688 C7APO2 57392934 IC50 = 1100 nM T50688 CZ2A0S 57392935 IC50 > 100000 nM T50688 CX16KB 57393324 IC50 = 45000 nM T50688 CR72PQ 57393920 IC50 = 4.4 nM T50688 C6EWL9 57394677 IC50 = 49000 nM T50688 C8T2ZJ 57395044 IC50 > 100000 nM T50688 C9F4OL 57398232 IC50 = 2000 nM T50688 C5OAB7 57398233 IC50 > 100000 nM T50688 CY39KP 57398234 IC50 > 100000 nM T50688 CODX48 57399879 IC50 = 2200 nM T50688 C93VSX 57399880 IC50 = 33000 nM T50688 C5WOZ3 57399881 IC50 = 31000 nM T50688 C9ZL5X 57400230 IC50 = 31000 nM T50688 CPZR79 57400272 IC50 = 60000 nM T50688 CJGQ60 57400873 IC50 = 6.3 nM T50688 CS2ZY1 57401658 IC50 = 1800 nM T50688 CG90KP 57403382 IC50 = 34000 nM T50688 C3CKA6 57403383 IC50 = 80000 nM T50688 C4OB6Z 57403384 IC50 = 2500 nM T50688 CKI4S8 57403776 IC50 = 2500 nM T50688 CR71ZG 59665343 IC50 > 10000 nM T50688 C31IUF 69863577 IC50 > 10000 nM T50688 CM2AD4 70696326 IC50 > 10000 nM T50688 CAF23V 71452640 IC50 > 200000 nM T50688 C23GSR 71459889 IC50 = 28000 nM T50688 C8EM7Y 71550913 IC50 > 10000 nM T50688 CU95LC 71574160 IC50 > 10000 nM T50688 COJ8Y4 71574161 IC50 > 10000 nM T50688 C8V4UB 71574356 IC50 > 10000 nM T50688 C9J7NH 71652207 IC50 = 42600 nM T50688 CLH52G 71654374 IC50 > 200000 nM T50688 C8GDV7 71654376 IC50 > 200000 nM T50688 CY29LR 71654530 IC50 > 200000 nM T50688 C3K6PT 71654532 IC50 > 200000 nM T50688 C3X7FP 71654534 IC50 = 1210 nM T50688 CCGP56 71654535 IC50 = 665 nM T50688 CZG3Y9 71654536 IC50 = 17600 nM T50688 C5D2OL 71698598 IC50 > 300000 nM T50688 CGYN76 71698686 IC50 > 300000 nM T50688 CD0Z5K 71698687 IC50 > 300000 nM T50688 C0DUT2 71698688 IC50 > 300000 nM T50688 C60JTA 71698689 IC50 > 300000 nM T50688 C35ZJV 71698690 IC50 > 300000 nM T50688 C9XSB5 71698770 IC50 = 78400 nM T50688 CRN95M 71698771 IC50 > 300000 nM T50688 C0LW4G 71698774 IC50 > 300000 nM T50688 CH26JR 71698775 IC50 = 16800 nM T50688 C0WR9F 71699124 IC50 = 14000 nM T50688 CZKL39 71699125 IC50 = 96000 nM T50688 C27TZK 71699126 IC50 = 55000 nM T50688 CD12FS 71699127 IC50 = 35000 nM T50688 CFN7Q4 71699199 IC50 = 12000 nM T50688 C7RTF0 71699200 IC50 = 4700 nM T50688 C8JE0W 71699201 IC50 = 2200 nM T50688 CRAG19 71699203 IC50 > 300000 nM T50688 CYAH23 71699286 IC50 > 300000 nM T50688 CM8E7F 71699287 IC50 = 25800 nM T50688 C9Y3DN 71699288 IC50 = 12800 nM T50688 C8B7QE 72949858 IC50 > 5000 nM T50688 CZ2P8U 73345565 IC50 = 30 nM T50688 CQAE56 73345568 IC50 = 220 nM T50688 CU1VZ5 73345570 IC50 = 60 nM T50688 CPT7S8 73345576 IC50 = 248 nM T50688 C0BJ1F 73345752 IC50 = 850 nM T50688 C9UD8K 73346937 Ki = 42000 nM T50688 CKG2D8 73346996 IC50 = 7970 nM T50688 C1Z4HB 73346997 IC50 > 200000 nM T50688 COP75R 73347022 IC50 = 1790 nM T50688 C5E4ZO 73347079 Ki = 13.7 nM T50688 CZ6Y9R 73347081 IC50 = 10 nM T50688 CZ35TD 73347085 IC50 = 352 nM T50688 CGM9F7 73347087 IC50 = 70 nM T50688 C89ENA 73347090 IC50 = 1 nM T50688 CN1A2D 73347092 IC50 = 400 nM T50688 C7IC1G 73347403 IC50 > 300000 nM T50688 CHLG51 73348500 IC50 = 150 nM T50688 CD1RB5 73348588 Ki = 4.8 nM T50688 CO9L2V 73348591 IC50 = 20 nM T50688 C43LWV 73348592 IC50 = 20 nM T50688 CM37AE 73348593 IC50 = 10 nM T50688 CT1RG5 73348594 IC50 = 40 nM T50688 CF1UL2 73348680 IC50 = 6000 nM T50688 C7Y3ZB 73348933 IC50 > 300000 nM T50688 CO15PX 73350083 IC50 = 200000 nM T50688 CU0GS5 73350084 IC50 = 385000 nM T50688 CH4VE1 73350172 Ki = 24.3 nM T50688 CQL5F8 73350174 Ki = 35 nM T50688 CQ5D7B 73350175 IC50 = 20 nM T50688 CJEH13 73350177 IC50 = 10 nM T50688 C20AJB 73350179 IC50 = 4 nM T50688 C19PJE 73350181 IC50 = 17 nM T50688 CRHV46 73351571 Ki = 58 nM T50688 C2F3YZ 73351673 IC50 = 210 nM T50688 CJA25I 73351674 IC50 = 150 nM T50688 C6NCQ1 73351675 IC50 = 50 nM T50688 C46ULG 73351676 IC50 = 150 nM T50688 C8B6NV 73351677 IC50 = 31 nM T50688 CIYV49 73351678 IC50 = 6 nM T50688 CY76LM 73353036 IC50 = 40500 nM T50688 CA6GB7 73353037 IC50 = 55300 nM T50688 CKW5X4 73353038 IC50 > 200000 nM T50688 CM94NF 73353043 IC50 = 32200 nM T50688 CR5HL8 73353062 Ki = 3300 nM T50688 CUE1A8 73353139 Ki = 8.5 nM T50688 C20FGN 73353141 IC50 = 40 nM T50688 CP6AJ3 73353143 IC50 = 30 nM T50688 CUPR57 73353147 IC50 = 30 nM T50688 C83RAM 73353150 IC50 = 29 nM T50688 CX47JD 73353160 IC50 = 120 nM T50688 C3QZ4W 73354557 IC50 = 82000 nM T50688 CUP3W4 73354558 IC50 = 9600 nM T50688 C6OX7Q 73354659 Ki = 58 nM T50688 CV3OI9 73354660 Ki = 9.3 nM T50688 CRY2K3 73354661 Ki = 26 nM T50688 CAJ27W 73354663 IC50 = 70 nM T50688 CT4A5S 73354664 IC50 = 90 nM T50688 C6XTP9 73354667 IC50 = 16 nM T50688 CZ1BL4 73354668 IC50 = 20 nM T50688 CC19KU 73356070 Ki = 75000 nM T50688 C1LZI2 73356125 IC50 = 11400 nM T50688 C8GVU2 73356136 IC50 = 26 nM T50688 C4EJK0 73356213 IC50 = 20 nM T50688 CH8G5C 73356216 IC50 = 120 nM T50688 CPG36Q 73356217 IC50 = 15 nM T50688 CD1S3N 73356221 IC50 = 50 nM T50688 CI07FE 90645591 IC50 = 947000 nM T50688 C8N6OE 90654504 IC50 > 10000 nM T50688 CRY16L 91930237 IC50 = 13 nM T50688 C3I5NZ 118709463 IC50 = 1.5 nM T50688 CY1IS6 118718872 IC50 = 10 nM T50688 CHD10T 118753906 IC50 = 220 nM T50688 CE7PC8 118753907 IC50 = 7900 nM T50688 CJX84K 122192536 IC50 = 320 nM T50688 CC57KE 122192704 IC50 = 79 nM T50688 C6PBW7 122192706 IC50 = 0.22 nM T50688 CGI3N9 122192708 IC50 = 0.96 nM T50688 CMU5L2 134132719 IC50 = 7600 nM T50688 CFO64Z 134132799 IC50 = 18800 nM T50688 C7FPL9 134135111 IC50 = 200 nM T50688 C3D0AC 134135726 IC50 = 7900 nM T50688 C4MU0L 134136847 IC50 = 6380 nM T50688 C1WMQ0 134137198 IC50 = 5400 nM T50688 CR2BO9 134137328 IC50 > 100000 nM T50688 CP5S6D 134137433 IC50 = 1330 nM T50688 CCN09H 134137713 IC50 > 100000 nM T50688 CSW65H 134138739 IC50 = 80 nM T50688 C7K5IZ 134139108 IC50 = 4010 nM T50688 CAP65B 134140093 IC50 > 100000 nM T50688 CB6SA2 134143022 IC50 = 370 nM T50688 CXNR60 134143874 IC50 = 520 nM T50688 C0UL6E 134146896 IC50 = 3290 nM T50688 CCGZ12 134147635 IC50 = 280 nM T50688 C5EL6I 134148127 IC50 = 24600 nM T50688 CZY3O5 134151321 IC50 = 2100 nM T50688 C4LV7R 134152693 IC50 = 1080 nM T50688 CIC9T4 134153084 IC50 = 3400 nM T50688 C3H8BS 134153267 IC50 = 1650 nM T50688 CMN95S 134153892 IC50 = 12700 nM T50688 C46ICN 134157552 IC50 = 12800 nM T50688 CJL87N 135949396 IC50 = 323 nM T50688 CSCN42 135983770 IC50 = 167 nM T50688 CR8K5L 135983772 IC50 = 6300 nM T50688 C1WEK2 136048740 IC50 = 20 nM T50688 CW4IZ6 136056116 IC50 = 400 nM T50688 CBVF84 136094924 IC50 = 3.8 nM T50688 C61NCW 136094926 IC50 = 150 nM T50688 CT1QN2 136224837 IC50 = 15300 nM T50688 CN8BW0 136224847 IC50 = 16000 nM T50688 C7KE9J 136224848 IC50 = 870 nM T50688 C7R1TS 136224849 IC50 = 890 nM T50688 CG24CQ 136224854 IC50 = 260 nM T50688 C4IE0Q 137028367 IC50 = 2.2 nM T50688 CL4K9J 137175047 IC50 = 55 nM T50688 CDQ5J6 137175053 IC50 = 1.8 nM T50688 CVAK07 137175055 IC50 = 1.53 nM T50688 C9C4AK 137175068 IC50 = 1.57 nM T50688 CACK48 137659180 IC50 = 2.3 nM T50688 C17RZG 155515221 IC50 = 5804 nM T50688 CHT1J6 155515540 IC50 > 1000 nM T50688 CQ5C4M 155516533 IC50 > 1000 nM T50688 CZY8F6 155520344 IC50 = 5028 nM T50688 C2GJ5V 155527654 IC50 > 10000 nM T50688 CPIL79 155528977 IC50 > 10000 nM T50688 CJZU81 155532583 IC50 > 10000 nM T50688 CJ7O2X 155534687 IC50 > 1000 nM T50688 CWF98D 155552156 IC50 > 1000 nM T50688 C80PGY 155563043 IC50 > 10000 nM T50688 CEF3T8 155563936 IC50 > 1000 nM T50688 C2M7AJ 15677293 IC50 = 30000 nM T50688 C5FR9J 44385169 IC50 = 43000 nM T50688 CXT94Y 44403730 IC50 = 14 nM T50688 D01XUU 9958398 IC50 = 8 nM T50688 D04BHL 177230 IC50 = 60 nM T50688 D04XTP 44322318 IC50 = 0.027 nM T50688 D05AGK 11743533 IC50 = 17 nM T50688 D06LHH 9805998 IC50 = 13 nM T50688 D06LKH 123811 IC50 = 120 nM T50688 D06LUT 44379110 IC50 = 3440 nM T50688 D07WDB 104802 IC50 = 76 nM T50688 D08RLR 9862322 IC50 = 67 nM T50688 D0A0KS 9851104 IC50 = 12000 nM T50688 D0B4JU 15409414 IC50 = 195 nM T50688 D0C8LA 9913833 IC50 = 9 nM T50688 D0H3UO 9984308 IC50 = 26 nM T50688 D0LV6B 130667 IC50 = 1700 nM T50688 D0M7KS 52942958 Ki = 110 nM T50688 D0O5OM 10742947 IC50 = 25000 nM T50688 D0R3CY 9952958 IC50 = 1200 nM T50688 D0S8DT 10324223 IC50 = 15 nM T50688 D0W5ZK 177364 IC50 = 12 nM T73482 D00OVU 24965990 Ki = 0.3981 nM T73482 D02RXG 6918287 Ki = 250 nM T73482 D06CKX 25195495 Ki = 0.3 nM T73482 D08SCL 46190695 IC50 = 1986 nM T73482 D0A7ZK 56944144 Ki = 2.512 nM T73482 D0FK6O 67116280 Ki = 1277 nM T73482 D0NN5A 25128145 Ki = 0.631 nM T73482 D06BTF 23727689 IC50 = 13 nM T73482 C91DAE 185394 Ki = 1300 nM T73482 CKN27R 645882 Ki > 15848.93 nM T73482 CW90GD 647720 Ki > 15848.93 nM T73482 CMQ23R 833756 Ki = 36 nM T73482 C5NO3B 855282 Ki > 15848.93 nM T73482 C1Q7FH 1034375 Ki = 1200 nM T73482 CCN92H 1207917 Ki = 6700 nM T73482 CEX5I0 1301005 IC50 = 21 nM T73482 CK8ZP2 1725151 IC50 > 10000 nM T73482 C7L9OX 1784975 IC50 > 10000 nM T73482 CZ0AJ2 2273636 IC50 > 10000 nM T73482 CDC1E3 2796191 Ki = 216 nM T73482 CC79VB 2860019 Ki = 6300 nM T73482 C4JH3Z 2870209 Ki = 30700 nM T73482 CV53JP 3119056 IC50 > 10000 nM T73482 CF8RB9 3119749 Ki = 2700 nM T73482 CG01OM 3213606 Ki > 15848.93 nM T73482 C4X9CJ 3213619 Ki > 15848.93 nM T73482 C4XGO6 3213626 Ki > 15848.93 nM T73482 C8WE7J 3213637 Ki > 15848.93 nM T73482 CL6KP4 3213649 Ki = 2511.89 nM T73482 C89CAQ 3213663 Ki > 15848.93 nM T73482 C7XRC5 3213671 Ki = 630.96 nM T73482 CA9E7M 3213679 Ki > 15848.93 nM T73482 CL7PN8 3213689 Ki = 1258.93 nM T73482 CFPR85 3213696 Ki = 794.33 nM T73482 CLX9G8 3213712 Ki > 15848.93 nM T73482 C9L6CG 3213744 Ki = 2511.89 nM T73482 CU8F4X 3213776 Ki = 2511.89 nM T73482 CJ93NE 3213793 Ki > 15848.93 nM T73482 CHS5V2 3213803 Ki > 15848.93 nM T73482 C4O1NG 3213835 Ki = 1995.26 nM T73482 C0IW7Z 3213904 Ki > 15848.93 nM T73482 C3XD5Z 3213915 Ki > 15848.93 nM T73482 CM2S1K 3213928 Ki = 794.33 nM T73482 C32UAN 3213941 Ki > 15848.93 nM T73482 C5R4LA 3213958 Ki > 15848.93 nM T73482 CYM81H 3213966 Ki = 1995.26 nM T73482 C8XAM0 3213992 Ki = 1000 nM T73482 CS0VF3 3214024 Ki = 3162.28 nM T73482 C2J1TB 3634416 Ki = 12000 nM T73482 C3O5WZ 5165198 Ki > 15848.93 nM T73482 C04ZBY 5218889 Ki = 800 nM T73482 CT23BD 6418917 Ki = 1100 nM T73482 CX1BS0 6859582 Ki = 7600 nM T73482 CTYZ64 9798764 Ki = 28 nM T73482 C7SN9C 9936247 IC50 = 5300 nM T73482 CR3LK5 9978819 Ki = 1995.26 nM T73482 C2ELV0 9978820 Ki = 1000 nM T73482 CK0F1B 10024157 Ki < 10000 nM T73482 C25NXP 10024223 Ki = 1000 nM T73482 CR4VC2 10044549 Ki = 2511.89 nM T73482 C8TZF9 10046197 Ki = 63.1 nM T73482 CO41BA 10046198 Ki > 5011.87 nM T73482 CER65W 10048862 Ki = 6.31 nM T73482 CC0V9S 10069829 Ki = 251.19 nM T73482 C8SHP4 10112247 IC50 > 10000 nM T73482 C7UL5G 10113123 Ki = 8 nM T73482 C8MS0F 10139334 IC50 = 18 nM T73482 C41SAC 10144095 IC50 = 52 nM T73482 C5CZ0J 10201185 Ki = 5.012 nM T73482 CV0Y8N 10204153 Ki = 1.1 nM T73482 CVN2Q8 10208109 IC50 = 17 nM T73482 C46ROY 10250023 Ki = 100 nM T73482 CTHA73 10278102 IC50 = 119 nM T73482 C69ZAN 10316124 Ki = 125.89 nM T73482 CYB3G4 10316232 Ki = 2511.89 nM T73482 CQNX31 10316508 Ki = 79.43 nM T73482 CWU80C 10337554 Ki = 398.11 nM T73482 CJSX37 10386388 Ki = 501.19 nM T73482 CZS4R9 10387337 Ki = 39.81 nM T73482 C8OF7V 10407090 Ki = 63.1 nM T73482 CA3E0X 10409682 IC50 > 10000 nM T73482 C4E9ZR 10433189 Ki = 501.19 nM T73482 C3LJ1G 10453273 Ki = 19.95 nM T73482 C5FBU7 10473775 Ki < 10000 nM T73482 CZ1J7A 10475401 IC50 > 10000 nM T73482 CX7M8O 10864072 IC50 = 127 nM T73482 C7OM4V 10864264 IC50 = 552 nM T73482 CBM0E3 10864538 IC50 = 19 nM T73482 CUPD25 10874416 IC50 = 9475 nM T73482 CV83MQ 10884498 IC50 = 5731 nM T73482 C8ZEK0 10906648 IC50 = 8425 nM T73482 CKV5W9 10918096 IC50 = 1460 nM T73482 C2VF5E 10918199 IC50 = 37 nM T73482 CVI01B 10929426 IC50 = 1906 nM T73482 C0MWO4 10939830 IC50 = 44 nM T73482 CVG1W4 10939855 IC50 = 1113 nM T73482 CKNF23 10951393 IC50 = 49 nM T73482 C4ZTW3 10951496 IC50 = 8 nM T73482 C8E5LJ 10962350 IC50 = 129 nM T73482 CE68HD 10983971 IC50 = 200 nM T73482 CADV49 10983972 IC50 = 2008 nM T73482 CRNI02 10994188 IC50 = 4274 nM T73482 CR9S3I 10994415 IC50 = 4771 nM T73482 C9KAL2 11016474 IC50 > 10000 nM T73482 C5W8OD 11016554 IC50 = 118 nM T73482 CC0IG1 11038242 IC50 = 1182 nM T73482 C4DX9L 11049263 IC50 = 1138 nM T73482 C3NL0R 11071336 IC50 = 45 nM T73482 CZF1P3 11071351 IC50 = 10000 nM T73482 C47DCI 11081493 IC50 = 268 nM T73482 C8RK9Q 11081686 IC50 = 3138 nM T73482 CF9D3V 11102681 IC50 > 10000 nM T73482 C5G1WK 11123332 IC50 = 4464 nM T73482 CGA21K 11146397 IC50 = 21 nM T73482 C16TCJ 11180190 Ki = 4.15 nM T73482 CM26ZQ 11734173 IC50 = 75 nM T73482 C6KE0W 11744563 Ki = 79.43 nM T73482 CZ0TU8 11812976 IC50 = 690 nM T73482 CM6A3U 11960895 Ki = 3 nM T73482 CHV29L 11960929 Ki = 8 nM T73482 CQD14I 12047522 IC50 > 10000 nM T73482 C5SR3I 12997499 IC50 > 10000 nM T73482 CXGJ06 15949515 Ki = 27 nM T73482 CDXM06 15949516 Ki = 86 nM T73482 CBF2K7 15949607 Ki = 40 nM T73482 C1EIU3 15949609 Ki = 130 nM T73482 CA3C9D 15949610 Ki = 28 nM T73482 C9V6OR 15949701 Ki = 500 nM T73482 C75IUA 15949702 Ki = 2300 nM T73482 CM61GE 15949703 Ki = 69 nM T73482 CJ4X8D 15993497 IC50 > 10000 nM T73482 C52SLH 16002587 Ki > 6309.57 nM T73482 C81AUJ 16046844 Ki = 79.43 nM T73482 C0BLR7 16048438 Ki = 954.99 nM T73482 C9RM2Y 16752731 IC50 = 6 nM T73482 CKH6B4 18592212 Ki = 7.943 nM T73482 CK7L1A 18592214 Ki > 2511.89 nM T73482 CT6ON8 18592216 Ki = 1995.26 nM T73482 CJBK87 20911062 IC50 = 3455 nM T73482 CQE54R 22599910 IC50 > 10000 nM T73482 CW7F3D 22599915 IC50 > 10000 nM T73482 CKL08P 22599923 IC50 > 10000 nM T73482 CIO42U 24737677 IC50 = 10 nM T73482 CBC56J 24748750 IC50 = 26 nM T73482 CH6TN9 24759955 IC50 = 17 nM T73482 CY3X7G 24760024 IC50 = 12 nM T73482 C4R8OV 24760087 IC50 = 29 nM T73482 C9B2DL 24760747 IC50 = 119 nM T73482 C43PRK 24760748 IC50 = 166 nM T73482 CB3TQ1 24808511 IC50 = 27 nM T73482 C1H3AN 24808514 Ki = 1.8 nM T73482 CK5LN1 24853522 IC50 = 7 nM T73482 COB2P9 24882716 Ki = 1.2 nM T73482 CB9SA1 24896566 Ki = 462 nM T73482 CZ9EQ2 24959177 IC50 = 40 nM T73482 C9MI0U 24959178 IC50 = 16 nM T73482 CJR42H 24959549 IC50 = 18 nM T73482 CY58BS 24959912 IC50 = 45 nM T73482 C50TAB 24960290 IC50 = 1066 nM T73482 C5UF2L 24960654 IC50 = 313 nM T73482 CTE96G 24961018 IC50 = 717 nM T73482 CUI6E1 24961746 IC50 = 20 nM T73482 C35DNF 24961747 IC50 = 32 nM T73482 C67KNQ 24962111 IC50 = 203 nM T73482 C57LWU 24962112 IC50 = 3902 nM T73482 CG43WT 24962115 IC50 = 459 nM T73482 CK9H5Y 24962833 IC50 = 431 nM T73482 CL6N8O 24962835 IC50 = 312 nM T73482 C95RZN 24964358 Ki = 1700 nM T73482 C9IUP7 24964576 Ki = 0.8 nM T73482 C38UID 24964578 Ki = 0.5 nM T73482 CYEP21 24964937 Ki = 0.3 nM T73482 C5I9DX 24965290 Ki = 0.2 nM T73482 C5SFH2 24965291 Ki = 0.3 nM T73482 CGP45R 24965643 Ki = 0.78 nM T73482 CSI6H9 24965645 Ki = 1.8 nM T73482 CFS95W 24968277 Ki = 0.7 nM T73482 CPQD14 24992490 IC50 = 3098 nM T73482 CTI38U 25060119 Ki = 94.5 nM T73482 CTX03U 25060120 Ki = 7250 nM T73482 C8XKP2 25060382 Ki = 3350 nM T73482 CXE52R 25060383 Ki = 1105 nM T73482 CD6CA4 25060384 Ki = 2975 nM T73482 C6L1VC 25060653 Ki = 236 nM T73482 C8DO2L 25060654 Ki = 273 nM T73482 CN7V6R 25060655 Ki = 833 nM T73482 C0K6WX 25060657 Ki = 1087 nM T73482 C5U9ZY 25060899 Ki = 1073 nM T73482 CDBQ73 25060900 Ki = 5150 nM T73482 C56RMG 25060902 Ki = 747 nM T73482 CMOS06 25063585 IC50 = 108 nM T73482 CF5AB2 25063587 IC50 = 358 nM T73482 CJY0H7 25063628 IC50 = 993 nM T73482 C7ZP8R 25063664 IC50 = 180 nM T73482 C9KY3W 25063665 IC50 = 1031 nM T73482 C39RAF 25063701 IC50 = 669 nM T73482 C15XCU 25127493 Ki = 1 nM T73482 CY5X1A 25204740 IC50 = 13 nM T73482 C03XSU 25225718 Ki = 720 nM T73482 CF5MV8 25809483 IC50 > 10000 nM T73482 C07DOP 26719840 IC50 = 31 nM T73482 CW2U6O 30560665 IC50 = 9191 nM T73482 CYL39Q 40924317 Ki = 6.31 nM T73482 C7IKX4 42604859 Ki = 900 nM T73482 CT13OI 44219762 Ki = 2 nM T73482 CI4BE6 44270595 EC50 > 1000000 nM T73482 CW30VO 44270596 EC50 > 1000000 nM T73482 C26BKD 44270597 EC50 > 1000000 nM T73482 C39TRO 44270625 EC50 > 1000000 nM T73482 C5PO4S 44270635 EC50 > 1000000 nM T73482 C87IBU 44270666 EC50 > 1000000 nM T73482 CMB6A1 44270673 EC50 > 1000000 nM T73482 C1OM8C 44270674 EC50 > 1000000 nM T73482 CZW96I 44270676 EC50 > 1000000 nM T73482 CQ56DO 44270709 EC50 > 1000000 nM T73482 C6GJW8 44359225 IC50 = 3600 nM T73482 CUPE16 44359281 IC50 = 3670 nM T73482 C68CJQ 44359282 IC50 = 1130 nM T73482 C9H4QW 44359283 IC50 > 10000 nM T73482 C5FKZ8 44359335 IC50 > 10000 nM T73482 CQP59C 44359365 IC50 = 5900 nM T73482 CIO8P6 44359366 IC50 > 10000 nM T73482 CE4FG6 44359367 IC50 = 3850 nM T73482 C7SO5Y 44359405 IC50 > 10000 nM T73482 CCG51L 44359415 IC50 = 5500 nM T73482 CX4C8G 44359451 IC50 > 10000 nM T73482 CSY89K 44359452 IC50 > 10000 nM T73482 CA31JT 44359467 IC50 > 10000 nM T73482 C9YK1T 44359482 IC50 > 10000 nM T73482 CFJI51 44359494 IC50 > 10000 nM T73482 COVU19 44359603 IC50 > 10000 nM T73482 CUQ13D 44359613 IC50 = 2300 nM T73482 CN73FK 44359637 IC50 = 7000 nM T73482 CR9E8A 44359650 IC50 > 10000 nM T73482 CN3HL7 44376980 Ki = 66069.34 nM T73482 C9QD1O 44376981 EC50 = 1380 nM T73482 CD62VI 44393273 Ki < 10000 nM T73482 C47MUJ 44393285 Ki < 5011.87 nM T73482 CT3U9Z 44393313 Ki = 125.89 nM T73482 C5QNK7 44393337 Ki < 10000 nM T73482 CIWP10 44393338 Ki < 10000 nM T73482 C81EBC 44393370 Ki = 501.19 nM T73482 C4X2QA 44393375 Ki < 10000 nM T73482 CH0UI9 44405008 EC50 = 5.7 nM T73482 CM1IS8 44454577 Ki = 10 nM T73482 CA39CP 44454599 Ki = 1400 nM T73482 C1BD8E 44454602 Ki = 2500 nM T73482 CR35JH 44454877 Ki = 15 nM T73482 C9OD7E 44454878 Ki = 2 nM T73482 CLRZ97 44454915 Ki = 0.7 nM T73482 CZG78N 44454916 Ki = 120 nM T73482 CYIO02 44454917 Ki = 3 nM T73482 CSLE81 44454943 Ki = 39 nM T73482 CWPB72 44454946 Ki = 9 nM T73482 C2RO9B 44454947 Ki = 49 nM T73482 C3I1LF 44463491 Ki = 1.995 nM T73482 CJY9N1 44555825 IC50 = 170 nM T73482 C92PMB 44555872 IC50 = 74 nM T73482 C2JT5F 44555974 IC50 = 85 nM T73482 C9UH1P 44555976 IC50 = 1677 nM T73482 C7P2VN 44555978 IC50 = 30 nM T73482 CJU9R7 44556023 IC50 = 94 nM T73482 C38KGZ 44556024 IC50 = 91 nM T73482 C3A8UM 44563904 IC50 = 19 nM T73482 C3IA9R 44563928 IC50 = 5 nM T73482 CCRY94 44563929 IC50 = 49 nM T73482 C5ASO0 44564034 IC50 = 3600 nM T73482 CR0T4G 44564035 IC50 = 731 nM T73482 CQ6Y4K 44564036 IC50 = 1565 nM T73482 CFA0L2 44564038 IC50 = 5300 nM T73482 C7R9DP 44574230 Ki = 9800 nM T73482 CZQ2N6 44574255 Ki = 930 nM T73482 C7IYO9 44574256 Ki = 63 nM T73482 C67JEM 44574257 Ki = 51 nM T73482 CUZK61 44580808 IC50 > 10000 nM T73482 C2R8YC 44580809 IC50 > 10000 nM T73482 C0LDE2 44580810 IC50 > 10000 nM T73482 CHIG04 44580825 IC50 = 2486 nM T73482 C6HQ2K 44580862 IC50 > 10000 nM T73482 CLP6W7 44580863 IC50 > 10000 nM T73482 C0BJI8 44580864 IC50 > 10000 nM T73482 CLKU70 44580865 IC50 = 886 nM T73482 C5INH4 44580886 IC50 = 4875 nM T73482 C2HT8N 44580887 IC50 = 1107 nM T73482 CUM2B9 44580888 IC50 = 888 nM T73482 C3FSE5 44580889 IC50 > 10000 nM T73482 CJ3HV2 44580912 IC50 = 1373 nM T73482 CEB05Y 44580913 IC50 = 2527 nM T73482 CC8D7N 44580914 IC50 = 1709 nM T73482 CY0A2T 44580945 IC50 = 17 nM T73482 CR8EL1 44580946 IC50 = 5 nM T73482 C2O6MI 44580947 IC50 = 12 nM T73482 CA36HG 44580948 IC50 = 6 nM T73482 CE4UV6 44580968 IC50 = 8 nM T73482 CVMS64 44580969 IC50 = 8 nM T73482 CNUF76 44581140 IC50 > 10000 nM T73482 CHZO78 44581141 IC50 > 10000 nM T73482 COUS06 44581168 IC50 > 10000 nM T73482 CNK67Y 44581169 IC50 > 10000 nM T73482 CZ03FY 44581170 IC50 > 10000 nM T73482 C41ZJE 44581171 IC50 > 10000 nM T73482 C97LXJ 44581172 IC50 > 10000 nM T73482 C6L7IF 44588748 Ki = 751 nM T73482 CDP50A 44588857 Ki = 1245 nM T73482 C1SYK4 44633765 Ki = 1584 nM T73482 CRM6C5 45259003 Ki = 10.5 nM T73482 C1QS3Y 45259004 Ki = 0.5 nM T73482 CH97EI 45375925 IC50 = 1950 nM T73482 CMRT28 45555989 IC50 = 6300 nM T73482 CB4O9P 46190694 Ki = 2700 nM T73482 C3KB9Q 46191662 IC50 = 3000 nM T73482 CRM02K 46191726 IC50 = 10000 nM T73482 CBGP17 46191727 IC50 = 10000 nM T73482 CJK6P2 46195690 Ki = 1000 nM T73482 CSJ27E 46204871 Ki = 2.2 nM T73482 CI34NU 46205522 Ki = 720 nM T73482 C2U1KF 46211807 Ki = 760 nM T73482 C0LQ6S 46211878 Ki = 900 nM T73482 C51BQE 46211883 Ki = 415 nM T73482 C48TNW 46211956 Ki = 2700 nM T73482 C21ICG 46212134 Ki = 965 nM T73482 C8R3SM 46212185 Ki = 910 nM T73482 CFV4Q2 46212296 Ki = 0.41 nM T73482 CHD1J4 46212539 Ki = 1030 nM T73482 CO7N9S 46212746 Ki = 4756 nM T73482 CT6F9H 46868664 Ki = 0.39 nM T73482 CNJR98 46868665 Ki = 6.2 nM T73482 CRK9B5 46868791 Ki = 4.1 nM T73482 C1KRZ6 46868793 Ki = 54 nM T73482 C7DH6F 46880346 IC50 = 10000 nM T73482 CP4C1B 46880347 IC50 = 63 nM T73482 C9Y3QE 46880348 IC50 = 1424 nM T73482 CMPE07 46880349 IC50 = 161 nM T73482 CJBC31 46880388 IC50 = 1919 nM T73482 CZ3C8T 46880389 IC50 = 402 nM T73482 C8ECV5 46880449 IC50 = 128 nM T73482 C29IMV 46880450 IC50 = 10000 nM T73482 C6JK5G 46880451 IC50 = 769 nM T73482 CFX08U 46883808 Ki = 1 nM T73482 C9C0FR 46883864 Ki = 12 nM T73482 CFL51W 46883865 Ki = 870 nM T73482 CR56NI 46883908 Ki = 0.4 nM T73482 CH5M1P 49793266 Ki = 8500 nM T73482 C51JSQ 49797987 Ki = 0.6 nM T73482 CS19WL 49797988 Ki = 0.9 nM T73482 CS9WK7 49798002 Ki = 10 nM T73482 C39KIH 49798003 Ki = 2 nM T73482 CR0C5N 49798004 Ki = 160 nM T73482 CNV6E4 49798005 Ki = 345 nM T73482 C3F0HR 49798028 Ki = 0.6 nM T73482 C72ADP 49798029 Ki = 7.6 nM T73482 C1X8TR 49798030 Ki = 0.4 nM T73482 C2BS3P 49805788 IC50 = 155 nM T73482 C0DKB7 50799599 Ki = 88 nM T73482 CS1O7E 52918933 Ki = 441 nM T73482 C51EGW 52942033 Ki > 15848.93 nM T73482 C65JKN 52944312 Ki > 15848.93 nM T73482 CFC12V 52944709 Ki > 15848.93 nM T73482 C9X3BC 52946457 Ki > 15848.93 nM T73482 CY9JU2 52948927 Ki > 15848.93 nM T73482 CJ4S2D 53242191 Ki = 288.4 nM T73482 CCZL67 53242213 Ki = 4 nM T73482 C8TC5B 53259112 Ki = 549.54 nM T73482 C68ERM 53259279 Ki = 1548.82 nM T73482 CK5CM6 53259467 Ki = 1424 nM T73482 C6U4FE 53259634 Ki = 58.88 nM T73482 CXKZ15 53259635 Ki = 18.62 nM T73482 C1HT7I 53259636 Ki = 275.42 nM T73482 C5E6TF 54576281 Ki = 4363 nM T73482 CI64JB 54579367 IC50 = 3784 nM T73482 CUG05N 54579583 IC50 = 2379 nM T73482 CAG6V1 54579585 IC50 > 10000 nM T73482 CLT6O5 54588789 IC50 = 998 nM T73482 C0OIE7 54751924 IC50 = 3000 nM T73482 C96GZT 54765113 IC50 = 6 nM T73482 CA0YR4 56659966 Ki = 10 nM T73482 CC6M4B 56663428 Ki = 501.19 nM T73482 CK76VA 56663429 Ki = 50.12 nM T73482 CU84LF 56670285 Ki = 125.89 nM T73482 C37HIB 56673796 Ki = 2511.89 nM T73482 C3CO2F 56673797 Ki = 6.31 nM T73482 CPT8J3 56673798 Ki = 1 nM T73482 CPE3R9 56680444 Ki = 398.11 nM T73482 C5TY1F 56680445 Ki = 7.943 nM T73482 CG6D7M 56680446 Ki = 39.81 nM T73482 CC0QF6 56683774 Ki = 0.1585 nM T73482 C35PTG 56683775 Ki = 0.1259 nM T73482 CW80YF 56943752 Ki = 30 nM T73482 CP5UD4 56944043 Ki = 2 nM T73482 C6F3VI 56944044 Ki = 137 nM T73482 CU87RH 56944045 Ki = 39 nM T73482 C67OXC 56944143 Ki = 3 nM T73482 C0BKG3 56944244 Ki = 32 nM T73482 C6GDX1 56944245 Ki = 39 nM T73482 CNY8F7 56944337 Ki = 121 nM T73482 C09WRF 56944429 Ki = 7 nM T73482 CAP79V 56944521 Ki = 43 nM T73482 C3SY9G 56944522 Ki = 9 nM T73482 CJ5T0W 56944620 Ki = 1 nM T73482 CX41CZ 56968452 Ki = 489.78 nM T73482 C6RH9Z 56970209 Ki = 812.83 nM T73482 CZQ5T1 56970417 Ki = 1621 nM T73482 C7I0LP 56970421 Ki = 21 nM T73482 C15GZB 56970625 Ki = 1445.44 nM T73482 CB4F3T 56970626 Ki = 371.54 nM T73482 CF7M3A 56970628 Ki = 660.69 nM T73482 CRV8S0 56970857 Ki = 1412.54 nM T73482 CDIO92 56970858 Ki = 512.86 nM T73482 CK9SF5 57388373 Ki > 2000 nM T73482 C56ORS 57388650 Ki = 106 nM T73482 CYQ43V 57388812 IC50 = 56.1 nM T73482 C1DF3J 57389725 IC50 = 3.22 nM T73482 CF08CS 57389801 IC50 = 5.54 nM T73482 CKDI91 57389883 IC50 = 119 nM T73482 C4FC6Z 57390049 IC50 = 9.06 nM T73482 C2LTP8 57390051 IC50 = 908 nM T73482 CB4CA1 57391006 IC50 = 1600 nM T73482 CAPD05 57392800 IC50 = 2300 nM T73482 C5WV2G 57396272 IC50 = 1600 nM T73482 C8DY2G 57398059 IC50 = 2600 nM T73482 C0K1PV 57403243 IC50 > 10000 nM T73482 C40IOT 57403244 IC50 = 1500 nM T73482 C9NHI3 58394291 IC50 = 10000 nM T73482 CXA3T8 58488153 Ki = 1 nM T73482 CI7U5V 60168601 IC50 = 5.4 nM T73482 CE9IM4 66733985 IC50 = 547 nM T73482 C8XNW4 67153780 IC50 = 53 nM T73482 CXQ94P 67153782 IC50 = 1426 nM T73482 C5FN3I 67209228 Ki = 778 nM T73482 C4PGT2 67209346 Ki = 29 nM T73482 CX2F3S 67209359 Ki = 274 nM T73482 CC2IT1 67209405 Ki = 20 nM T73482 CSQ3W1 67209426 Ki = 2667 nM T73482 CB7W0G 67209575 Ki = 970 nM T73482 C69PEQ 67209610 Ki = 800 nM T73482 C0C4JF 67209817 Ki = 63 nM T73482 CU5C8L 67251476 Ki = 1479.11 nM T73482 CC6X2O 67252378 Ki = 9.12 nM T73482 C4KC6Q 67281908 Ki = 3 nM T73482 CZ4L7E 67282493 Ki = 12 nM T73482 C3Q6ZA 67282848 Ki = 14 nM T73482 C4R1IH 67283149 Ki = 6 nM T73482 C0S7IR 67289227 Ki = 776.25 nM T73482 C15EQH 67380581 Ki = 3600 nM T73482 CH6EW0 67473922 Ki = 224 nM T73482 C1I7OW 67473934 Ki = 1016 nM T73482 CK18IT 67473935 Ki = 391 nM T73482 C2VD6Q 67473936 Ki = 1581 nM T73482 C42FLR 67473937 Ki = 138 nM T73482 CK1Q3V 67473938 Ki = 124 nM T73482 C2D4VM 67980311 Ki = 106 nM T73482 C0U9GM 67980666 Ki = 1068 nM T73482 CEVG41 68058790 Ki = 938 nM T73482 CDQ31I 68058793 Ki = 73 nM T73482 CTL92R 68083077 Ki = 81 nM T73482 CW8FR2 69080080 IC50 = 1950 nM T73482 CUIC59 69080156 IC50 = 25 nM T73482 CCB80U 69080186 IC50 = 107 nM T73482 CV4NO2 69080188 IC50 = 121 nM T73482 CN5H2Z 69080268 IC50 = 22 nM T73482 C58BVC 69080890 IC50 = 264 nM T73482 CE4I3Q 69080992 IC50 = 216 nM T73482 CJ7VG2 69081444 IC50 = 141 nM T73482 C49PMK 69081570 IC50 = 9 nM T73482 CNJ7K2 69081619 IC50 = 191 nM T73482 C4IW9J 69081640 IC50 = 65 nM T73482 CU4Z7I 69081642 IC50 = 40 nM T73482 CY0K1B 69081717 IC50 = 284 nM T73482 CD8RY3 69081742 IC50 = 19 nM T73482 CI3M2O 69081821 IC50 = 142 nM T73482 CSX60D 69081873 IC50 = 65 nM T73482 C30PMS 69081899 IC50 = 1407 nM T73482 CJI32G 69081964 IC50 = 16 nM T73482 CIN3O2 69082001 IC50 = 619 nM T73482 C3RDA0 69082236 IC50 = 75 nM T73482 C0QY5T 69082267 IC50 = 3486 nM T73482 CUW42P 69082306 IC50 = 77 nM T73482 C72OGM 69082473 IC50 = 4385 nM T73482 CJ93CT 69082475 IC50 = 32 nM T73482 C8L6DC 69082510 IC50 = 45 nM T73482 C6QB2K 69082516 IC50 = 3 nM T73482 CHS32F 69082545 IC50 = 3380 nM T73482 C95XAQ 69082595 IC50 = 899 nM T73482 CNK12W 69082599 IC50 = 2680 nM T73482 CW6MR8 69082645 IC50 = 44 nM T73482 C61XNT 69082665 IC50 = 4883 nM T73482 CD5HB2 69082678 IC50 = 177 nM T73482 CV94BF 69082681 IC50 = 154 nM T73482 CLX8D3 69082742 IC50 = 225 nM T73482 CJ45VT 69082766 IC50 = 412 nM T73482 CB70SA 69082817 IC50 = 136 nM T73482 COE39Z 69082854 IC50 = 927 nM T73482 C96STB 69082926 IC50 = 54 nM T73482 C6PR7O 69083435 IC50 = 193 nM T73482 CQ1IK8 69083745 IC50 = 1249 nM T73482 CPLG25 69083777 IC50 = 2 nM T73482 CJ6A5F 69084016 IC50 = 299 nM T73482 CKH1J6 69084057 IC50 = 1270 nM T73482 C3WL1H 69084118 IC50 = 4 nM T73482 C4E9VH 69084152 IC50 = 675 nM T73482 CT2NK9 69084345 IC50 = 44 nM T73482 CQPA54 69084621 IC50 = 1800 nM T73482 C2P3LC 69085010 IC50 = 724 nM T73482 C4NU5T 69085032 IC50 = 330 nM T73482 C4SXT9 69085047 IC50 = 14 nM T73482 C8T0RS 69085151 IC50 = 5 nM T73482 C4RU6S 69085189 IC50 = 14 nM T73482 CA4U1J 69085230 IC50 = 169 nM T73482 C9WX0M 69085295 IC50 = 1086 nM T73482 C4LM9J 69085642 IC50 = 531 nM T73482 CV76IC 69085689 IC50 = 550 nM T73482 C19PIM 69085726 IC50 = 34 nM T73482 C0Z1PN 69915149 Ki = 200 nM T73482 CP0N1Y 69915187 Ki = 52 nM T73482 C4I6UA 69915196 Ki = 4 nM T73482 C81MDP 69932186 Ki = 33 nM T73482 CA47RE 70169296 IC50 = 4364 nM T73482 CHS9N3 70681618 IC50 < 1 nM T73482 CB2QP1 70681619 IC50 = 8 nM T73482 C4NVY5 70681620 IC50 = 14 nM T73482 CUS92R 70683739 IC50 = 5 nM T73482 CM41XZ 70683740 IC50 = 6 nM T73482 CAU6W8 70683741 IC50 = 0.8 nM T73482 CDL7J3 70683742 IC50 = 145 nM T73482 C86KLO 70683743 IC50 > 2000 nM T73482 C4BOP2 70683744 IC50 = 390 nM T73482 C8PTI4 70685886 IC50 = 15 nM T73482 CWJ49Q 70685887 IC50 = 7 nM T73482 C5X8YM 70685888 IC50 = 6 nM T73482 C9O3RU 70685889 IC50 = 40 nM T73482 CFB9I0 70685890 IC50 = 1 nM T73482 CR7O0Q 70685891 IC50 = 121 nM T73482 C8YIC1 70685892 IC50 = 7 nM T73482 C6B1TJ 70687123 IC50 = 280 nM T73482 C80BKR 70687129 IC50 = 2500 nM T73482 C8G0AY 70688011 IC50 = 9 nM T73482 CTM9C1 70688012 IC50 = 2 nM T73482 C1IZ0S 70690040 IC50 = 4 nM T73482 CGA5E6 70690041 IC50 = 2 nM T73482 CCQR15 70690042 IC50 = 0.8 nM T73482 C3BRE9 70692193 IC50 = 3 nM T73482 CVT4S0 70692194 IC50 = 146 nM T73482 C0VL4I 70692195 IC50 = 27 nM T73482 C36FDI 70694255 IC50 = 2 nM T73482 CG4N1Z 70694256 IC50 = 12 nM T73482 CA58UO 70694257 IC50 = 6 nM T73482 C7UW0O 70696349 IC50 = 13 nM T73482 C0J2OK 70696350 IC50 = 10 nM T73482 CIPR26 70696351 IC50 = 2 nM T73482 CB3VS5 70816735 Ki > 4000 nM T73482 CWHM94 70816905 Ki = 175 nM T73482 C4RMS1 70817021 Ki = 2287 nM T73482 C94LXI 70817051 Ki = 783 nM T73482 CSCO94 70817059 Ki = 357 nM T73482 C7DO1N 70817239 Ki = 3 nM T73482 C6L7FH 70817382 Ki = 8 nM T73482 CTQ7C0 70818984 Ki = 660 nM T73482 CY03PE 70856594 Ki = 109 nM T73482 C7Q8ST 71522361 Ki = 1.1 nM T73482 C34TKD 71526207 Ki = 569 nM T73482 C2RO5Y 71526208 IC50 = 8400 nM T73482 CZ7JD6 71527494 Ki = 0.3 nM T73482 CE9SK3 71543409 Ki = 829 nM T73482 CR01NT 71555054 Ki = 4100 nM T73482 CTS09B 71579478 IC50 = 344 nM T73482 C12KAY 71579479 IC50 = 90 nM T73482 CJN41M 71580771 IC50 = 10000 nM T73482 C3QZ7D 71580772 IC50 = 10000 nM T73482 CV8N1K 71580773 IC50 = 10000 nM T73482 C4C9IF 71580858 IC50 = 10000 nM T73482 CX6G8Z 71580859 IC50 = 10000 nM T73482 CW7K4I 71580860 IC50 = 4171 nM T73482 CDC7T6 71580861 IC50 = 150 nM T73482 CQ2KC8 71580862 IC50 = 283 nM T73482 CL26RK 71580946 IC50 = 134 nM T73482 C9FIW3 71580947 IC50 = 3980 nM T73482 CAS05K 71580948 IC50 = 537 nM T73482 C0ND2T 71580949 IC50 = 10000 nM T73482 C5WL4U 71580950 IC50 = 492 nM T73482 C1NL7J 71624633 Ki = 900 nM T73482 CWAY56 71716523 IC50 = 1645 nM T73482 C1NP2M 72543760 IC50 = 1.25 nM T73482 CHU29Z 72699430 IC50 = 10.6 nM T73482 C1HMV0 72699854 IC50 = 1.07 nM T73482 CBF7O2 72699855 IC50 = 1.82 nM T73482 CKL84I 72699856 IC50 = 1.84 nM T73482 C1RY5X 72699949 IC50 = 1.26 nM T73482 C3I2OZ 72699950 IC50 = 0.82 nM T73482 CC70PO 72699951 IC50 = 3.06 nM T73482 C6HEI3 72700096 IC50 = 3.58 nM T73482 CH04OF 72700180 IC50 = 1.81 nM T73482 C5BKV3 72700181 IC50 = 2.01 nM T73482 CYJ2T4 72700265 IC50 = 1.58 nM T73482 CO7BI8 72700266 IC50 = 1.4 nM T73482 CL1U4W 72700267 IC50 = 2.45 nM T73482 CJN5K0 72700268 IC50 = 6.15 nM T73482 CZ8K4T 72700362 IC50 = 9.45 nM T73482 C7BY8D 72700363 IC50 = 1.93 nM T73482 CHCM80 72700366 IC50 = 14.7 nM T73482 CZDM79 72700457 IC50 = 4.39 nM T73482 CTLC87 72700458 IC50 = 1.9 nM T73482 CSWL87 72700459 IC50 = 86.6 nM T73482 CPV92B 72700460 IC50 = 1.1 nM T73482 C5JT0D 72700462 IC50 = 1.26 nM T73482 CWZ0T6 72700543 IC50 = 0.767 nM T73482 CP8G5V 72700544 IC50 = 4.39 nM T73482 COSK78 72700626 IC50 = 1.62 nM T73482 C68GDU 72700698 IC50 = 3.24 nM T73482 CMP5F9 72703893 IC50 < 10000 nM T73482 C7ZAH6 72703894 IC50 < 10000 nM T73482 CW3NX0 72704097 Ki = 20.42 nM T73482 CEY4I0 72704098 Ki = 1318.26 nM T73482 COTU10 72704099 Ki = 707.95 nM T73482 CGV76N 72704100 Ki = 758.58 nM T73482 CBE48L 72707143 Ki = 19.95 nM T73482 CO0U6I 72720554 Ki = 15.85 nM T73482 CVO7T2 72720555 Ki = 1 nM T73482 CD8Z5T 72720556 Ki = 39.81 nM T73482 CXG47B 72720982 Ki = 1.259 nM T73482 CBW93F 72721081 Ki = 63.1 nM T73482 CHN0B5 72721178 Ki = 316.23 nM T73482 C4OD7F 72721280 Ki = 25.12 nM T73482 C41JEL 72721380 Ki = 6.31 nM T73482 C50CDB 72721381 Ki = 63.1 nM T73482 CG8PX4 72721795 Ki = 50.12 nM T73482 CLD36Y 72721986 Ki = 25.12 nM T73482 C3JBG7 72721987 Ki = 1.995 nM T73482 C82DJS 72722084 Ki = 0.3981 nM T73482 CYC8U4 72722088 Ki = 12.59 nM T73482 C46UAR 72722089 Ki = 2.512 nM T73482 C6Q3OM 72725148 Ki = 1900 nM T73482 C3R1AC 72725149 Ki = 65000 nM T73482 C8DAZ2 73346054 IC50 = 5 nM T73482 C2C7BU 73347449 IC50 = 16 nM T73482 CO7CY6 73347581 IC50 = 10 nM T73482 CB8F6U 73348981 IC50 = 72 nM T73482 C8KLQ1 73350080 EC50 = 1340 nM T73482 CGZ7E4 73352057 IC50 = 378 nM T73482 CA9H1U 73353033 EC50 > 1000000 nM T73482 CJ4N5L 73353523 IC50 = 30 nM T73482 CB63NL 73356120 EC50 > 1000000 nM T73482 CIC73L 73356574 IC50 = 17 nM T73482 CH7S6O 73356708 Ki = 1400 nM T73482 C15PYW 73673014 Ki = 56 nM T73482 C34LXD 74221626 Ki = 757 nM T73482 C6M7RX 74221720 Ki = 572 nM T73482 CN53AG 74221903 Ki = 2517 nM T73482 CAIZ14 74221990 Ki = 1662 nM T73482 C7SZG6 74222158 Ki = 114 nM T73482 C6J9LF 74222159 Ki = 3568 nM T73482 C5J9EI 74222241 Ki = 1170 nM T73482 CZA0I9 74222326 Ki = 519 nM T73482 C07NHS 74222327 Ki = 1155 nM T73482 CGI5K2 74222402 Ki = 594 nM T73482 CZO3V4 74222406 Ki = 1611 nM T73482 CL15XT 74222492 Ki = 790 nM T73482 CA1N8P 74222754 Ki = 5765 nM T73482 CP9U0C 74222941 Ki = 1128 nM T73482 CX5L0W 76072813 Ki = 287 nM T73482 CF5Z2M 76310080 Ki = 3550 nM T73482 C28XZD 76310131 EC50 = 1130 nM T73482 CE5A0O 76310198 EC50 = 1040 nM T73482 CFS27O 76310208 EC50 = 526 nM T73482 CJO7X0 76310209 EC50 = 535 nM T73482 CE92OC 76310210 EC50 = 1560 nM T73482 CG3RK5 76310211 EC50 = 3070 nM T73482 CLY90X 76310431 IC50 > 10000 nM T73482 C6W4YC 76310456 IC50 = 1150 nM T73482 CT20QS 76313798 EC50 = 5700 nM T73482 C9V7HM 76313820 EC50 = 144 nM T73482 C07WGU 76313901 EC50 = 1360 nM T73482 C5ZE9C 76317346 EC50 = 1910 nM T73482 CEVZ91 76317683 IC50 = 17 nM T73482 C6CFQ9 76321148 EC50 = 2480 nM T73482 CP8M6Z 76321165 EC50 = 739 nM T73482 CM5HF7 76321386 IC50 = 2649 nM T73482 C9DZN3 76324691 EC50 = 1900 nM T73482 C1XSG9 76324989 IC50 = 32 nM T73482 CB3K9C 76328274 EC50 = 1370 nM T73482 CR6W3T 76328275 EC50 = 143 nM T73482 C6I7AK 76328558 IC50 = 14 nM T73482 C3O9LC 76331924 EC50 = 78.9 nM T73482 CRUK21 76331925 EC50 = 212 nM T73482 CVR8O9 76331964 EC50 = 865 nM T73482 CC9AR4 76332010 EC50 = 493 nM T73482 C54AVH 76332217 IC50 = 1590 nM T73482 C48LQC 76332218 IC50 = 2423 nM T73482 CNK25I 76332219 IC50 = 9704 nM T73482 C0ZN3F 76332238 IC50 = 537 nM T73482 CA1Z7X 76335540 EC50 = 1200 nM T73482 CV8NM6 76335605 EC50 = 3230 nM T73482 CVK6J7 76335606 EC50 = 422 nM T73482 CS2Y8O 76335607 EC50 = 3070 nM T73482 C2RVH7 76335608 EC50 = 3060 nM T73482 CRQ65T 76335879 IC50 > 10000 nM T73482 C0N3ZY 76534175 Ki = 391 nM T73482 CJG45W 76900605 Ki = 310 nM T73482 CXS7B6 77107594 Ki = 1.3 nM T73482 CVK3R4 78324905 Ki = 140 nM T73482 CZ8FN7 86267288 IC50 = 397 nM T73482 CEQ2V4 86269345 IC50 = 82 nM T73482 C9WI2E 86271116 Ki = 8 nM T73482 C9PVK1 86276237 IC50 = 18 nM T73482 CF4QX9 86278359 Ki = 800 nM T73482 C0PUY4 86291876 Ki = 64 nM T73482 CK6WQ1 86291877 Ki = 59 nM T73482 CHB7U8 86291879 IC50 = 828 nM T73482 CR32FQ 86292273 Ki = 120 nM T73482 CU0NT8 86298249 Ki = 130 nM T73482 CH4XK1 86302551 Ki = 0.5 nM T73482 CL7C5E 86302552 Ki = 0.9 nM T73482 C47MVU 86695644 IC50 = 14 nM T73482 CK9I5Y 89789751 IC50 = 3 nM T73482 C39TXO 89789760 IC50 = 2 nM T73482 C9I6NQ 89789762 IC50 = 264 nM T73482 C8S7BC 89789778 IC50 = 81 nM T73482 C0M7SQ 89789795 IC50 = 86 nM T73482 CERC67 89789843 IC50 = 20 nM T73482 CY9O3G 90405964 Ki = 12 nM T73482 C2WGJ3 90654337 Ki = 75 nM T73482 C8YE0S 90654338 Ki = 0.56 nM T73482 CZIE39 90654339 Ki = 470 nM T73482 C6TGU4 90654340 Ki = 17 nM T73482 CK38IX 90654341 Ki = 135 nM T73482 CL7KM1 90654342 Ki = 27 nM T73482 CFQS07 90654343 IC50 = 83 nM T73482 C8APK1 90654344 Ki = 26 nM T73482 C71YVR 90654345 Ki = 24 nM T73482 C2E5MT 90654346 Ki = 866 nM T73482 CPKH23 90654347 Ki = 211 nM T73482 CN7CX5 90654348 Ki = 18 nM T73482 CF0T9O 90654349 Ki = 76 nM T73482 C37MYP 90654350 Ki = 339 nM T73482 CJT36M 90654351 Ki = 108 nM T73482 CJ0Z5H 90656176 Ki = 0.7 nM T73482 CCW7S2 90656177 Ki = 0.3 nM T73482 C3EN1D 90656178 Ki = 2 nM T73482 CRK0W5 90656179 Ki = 4.5 nM T73482 CDN8Y4 90656180 Ki = 1.8 nM T73482 CJUS40 90656181 Ki = 1.8 nM T73482 CPSI06 90656182 Ki = 0.4 nM T73482 C8ZFG3 91801202 Ki = 1.585 nM T73482 C0DFT8 91809243 Ki = 166 nM T73482 CP0CE9 91810287 Ki = 140 nM T73482 CXO4N6 117668910 Ki = 430 nM T73482 C4HZ0N 117857721 IC50 = 3840 nM T73482 CJA8G5 117859490 IC50 > 10000 nM T73482 C1O2AH 117859572 IC50 = 21 nM T73482 C0CPN6 117859931 IC50 = 330 nM T73482 CZ20RX 118020300 IC50 = 10.1 nM T73482 C2Z1IN 118020504 IC50 = 61.5 nM T73482 CNI86H 118020539 IC50 = 245 nM T73482 CNKV57 118167452 Ki = 324 nM T73482 CSA7U9 118175269 Ki = 834 nM T73482 C72NVT 118175279 Ki = 6.3 nM T73482 CDAS04 118180165 Ki = 12 nM T73482 CK90HX 118435993 Ki = 1887 nM T73482 CF52MN 118715605 Ki = 2400 nM T73482 C4VR8L 118715606 IC50 > 10000 nM T73482 CG8MX4 118715607 IC50 > 10000 nM T73482 C1WKZ9 118715608 IC50 > 10000 nM T73482 CW4Z5M 118715609 IC50 = 4650 nM T73482 CN36LS 118715610 IC50 = 15000 nM T73482 C51JPK 118715611 IC50 = 10000 nM T73482 C1J2CY 118715612 Ki = 1500 nM T73482 CN14EP 118715613 Ki = 930 nM T73482 CNWA97 118716929 Ki > 10000 nM T73482 C3NW1S 118716930 Ki > 10000 nM T73482 CI3TK2 118716931 Ki = 4161 nM T73482 C5WRI1 118716932 Ki = 7.2 nM T73482 C5OQ4Y 118716933 Ki = 2994 nM T73482 C36PCB 118716934 Ki = 7535 nM T73482 CCT4Y0 118716935 Ki = 10000 nM T73482 CWJ69M 118716936 Ki = 6841 nM T73482 C9YEL0 118716937 Ki > 10000 nM T73482 CG5R1B 118716938 Ki = 5538 nM T73482 CHK4C7 118716939 Ki > 10000 nM T73482 CG75OB 118716940 Ki = 747 nM T73482 CG52QK 118716941 Ki = 772 nM T73482 C0QS6Y 118716942 Ki = 206 nM T73482 C10SEV 118716943 Ki = 1425 nM T73482 CAF89K 118716944 Ki = 291 nM T73482 C60JTD 118716945 Ki = 832 nM T73482 C2U1BX 118716946 Ki = 505 nM T73482 C83SPX 118716947 Ki = 106 nM T73482 C5ELB1 118716948 Ki = 103 nM T73482 C37UXI 118726303 Ki = 5.5 nM T73482 CFN4Y7 118726304 Ki = 106 nM T73482 C1Z7TR 118726305 Ki = 9 nM T73482 CX51TS 118726306 Ki = 13 nM T73482 CLQ34R 118726309 Ki = 470 nM T73482 CZ3OB5 118726310 Ki = 1100 nM T73482 C9WN2G 118726311 Ki = 510 nM T73482 CHM76O 118726312 Ki = 19000 nM T73482 C5S4RU 118726313 Ki = 1360 nM T73482 CS09EU 118726314 Ki = 1200 nM T73482 CN2KE3 118731950 IC50 = 3960 nM T73482 CF4QD0 118731951 IC50 = 7030 nM T73482 CYNB60 118731952 IC50 = 1980 nM T73482 C0VU1B 118731953 IC50 = 5780 nM T73482 CH8T0S 118731954 IC50 = 2400 nM T73482 C7KX2R 118731955 IC50 = 8720 nM T73482 CWA05F 118731956 IC50 = 3620 nM T73482 CC3PT6 118731957 IC50 = 467 nM T73482 CXEO47 118731958 IC50 = 1200 nM T73482 CTY98B 118736949 Ki = 12 nM T73482 C19HQW 118736950 Ki = 37 nM T73482 CRJ9L8 118736951 Ki = 14000 nM T73482 C82NQB 118736952 Ki = 57 nM T73482 CVO72M 118736953 Ki = 49 nM T73482 CWH08B 118736954 Ki = 470 nM T73482 CLAR49 118736955 Ki = 39 nM T73482 C3G6VD 118736956 Ki = 350 nM T73482 CCK3A9 118736957 Ki = 1400 nM T73482 CYBN01 118736958 Ki = 360 nM T73482 CLNY63 118736959 IC50 = 10000 nM T73482 CNU4D7 118736960 IC50 = 7100 nM T73482 CKFZ15 118736961 IC50 = 3300 nM T73482 COPD90 118736962 IC50 > 10000 nM T73482 CJ3VD1 118736963 IC50 > 10000 nM T73482 CMRB20 121231398 Ki = 393 nM T73482 CYHP86 122179999 Ki > 2000 nM T73482 CI3Q9N 122180000 Ki > 2000 nM T73482 CND0S5 122180001 Ki = 171 nM T73482 C0T3SD 122180002 Ki = 2491 nM T73482 C6CG5E 122180317 Ki = 6850 nM T73482 CQR14H 122180318 Ki = 5300 nM T73482 CE36GC 122180319 Ki > 10000 nM T73482 CVL0Q7 122180320 Ki > 10000 nM T73482 CW8H2J 122180321 Ki > 10000 nM T73482 CS1JC7 122180322 Ki = 1398 nM T73482 C6FVZ0 122180323 Ki = 925 nM T73482 CX9JG0 122180324 Ki = 267 nM T73482 CQU2H9 122180325 Ki = 765 nM T73482 CA5CP8 122180326 Ki = 1320 nM T73482 C6CAZ0 122180327 Ki > 10000 nM T73482 CRVB56 122180328 Ki > 10000 nM T73482 CAL3T2 122180329 Ki = 623 nM T73482 C3OJS0 122180330 Ki = 471 nM T73482 C4YIX5 122180331 Ki = 1800 nM T73482 C2DZ3Y 122180332 Ki = 3300 nM T73482 C0W3JG 122180333 Ki > 10000 nM T73482 C6EF1H 122180334 Ki = 557 nM T73482 C8SD7F 122180335 Ki = 257 nM T73482 C2WV9G 122180336 Ki = 1640 nM T73482 CJ1AP3 122180337 Ki = 2280 nM T73482 CBN0J2 122180338 Ki = 1960 nM T73482 CEA80S 122180339 Ki = 5780 nM T73482 CTG4B2 122180340 Ki = 3650 nM T73482 C6Y0JD 122180341 Ki = 680 nM T73482 CTCN25 122180342 Ki = 3090 nM T73482 C35BFD 122180343 Ki = 346 nM T73482 C80QZN 122180344 Ki = 5750 nM T73482 C6YIR4 122180345 Ki = 4630 nM T73482 CO1AK6 122184039 Ki = 0.06 nM T73482 C5XOD3 122184040 Ki = 23 nM T73482 CAYV10 122184041 IC50 = 259 nM T73482 CUWG52 122184042 Ki = 19 nM T73482 CTL34Z 122184043 Ki = 10 nM T73482 CVRO25 122184044 Ki = 12 nM T73482 C3WUY1 122184045 Ki = 4 nM T73482 C9HF4M 122191823 EC50 = 5227 nM T73482 CBI0X1 122191829 EC50 = 9248 nM T73482 CQ8FE7 122192247 EC50 = 6134 nM T73482 C5YRQ9 122192248 EC50 = 5720 nM T73482 CMX26J 122192250 EC50 = 2750 nM T73482 C4TX5S 122195752 Ki = 7 nM T73482 CD57NR 127027859 Ki = 34 nM T73482 CM91FC 127037650 IC50 = 16 nM T73482 CBT18A 127037651 IC50 = 45 nM T73482 CLD41N 127037996 IC50 = 2.7 nM T73482 C8INE9 127038060 IC50 = 16 nM T73482 CC3T8J 127038061 IC50 = 23 nM T73482 CJ03FI 127038062 IC50 = 3.5 nM T73482 CACI97 127038343 IC50 = 60 nM T73482 C4P7YM 127038416 IC50 = 33 nM T73482 C54FRL 127038812 IC50 = 64 nM T73482 CV6QR8 127038813 IC50 = 3.4 nM T73482 CRE04H 127038817 IC50 = 13 nM T73482 C71SOB 127038818 IC50 = 22 nM T73482 CRY01S 127038819 IC50 = 111 nM T73482 CSHM50 127038820 IC50 = 9.1 nM T73482 CNG1V0 127038821 IC50 = 11 nM T73482 CW47SG 127038822 IC50 = 8.3 nM T73482 CV8Z7T 127039127 IC50 = 3.8 nM T73482 CVOW03 127039128 IC50 = 26 nM T73482 C5IX1B 127039129 IC50 = 33 nM T73482 C1YUH6 127039134 IC50 = 11 nM T73482 C1NZ6H 127039135 IC50 = 17 nM T73482 CIBD78 127040414 IC50 = 28 nM T73482 COM28D 127040734 IC50 = 131 nM T73482 C37QEO 127040735 IC50 = 28 nM T73482 C6DEH8 127040736 IC50 = 108 nM T73482 CAX2I9 127040737 IC50 = 8.5 nM T73482 CTW7A2 127041999 Ki = 398.11 nM T73482 C07JPS 127042658 IC50 = 35 nM T73482 CX46KS 129093666 Ki = 1.96 nM T73482 CMZL51 129093667 Ki = 12.5 nM T73482 CP4TZ9 129093668 Ki = 6.21 nM T73482 CQ3I9T 129093669 Ki = 7.3 nM T73482 C5ZB7M 129093671 Ki = 13.9 nM T73482 C7M4SR 129093672 Ki = 12.1 nM T73482 C10DMA 129093673 Ki = 4.16 nM T73482 C4ABF5 129093675 Ki = 5.94 nM T73482 C4SU9L 129093829 Ki = 12 nM T73482 C40IXC 129093915 Ki = 2.1 nM T73482 C37OWP 129093916 Ki = 5.13 nM T73482 C9WTZ8 129093917 Ki = 3.47 nM T73482 CSB23A 129093918 Ki = 2.27 nM T73482 C3BI6O 129093944 Ki = 2.98 nM T73482 C8OD1A 129093945 Ki = 5.85 nM T73482 C1NF8H 129093946 Ki = 1.7 nM T73482 CDH9X8 129093947 Ki = 2.05 nM T73482 CV37XJ 129093951 Ki = 1.93 nM T73482 CRA76C 129093952 Ki = 7.6 nM T73482 CET1F7 129093953 Ki = 4.05 nM T73482 C2LWQ1 129093954 Ki = 2.07 nM T73482 CJB3M8 129093969 Ki = 6.19 nM T73482 CKL03Y 129093972 Ki = 12.6 nM T73482 CHB4I5 129093973 Ki = 1.81 nM T73482 C59FVA 129093974 Ki = 5.05 nM T73482 CSFT64 132537576 Ki = 1.36 nM T73482 CU58RD 135314438 Ki = 2.06 nM T73482 C9RA0Q 135314513 Ki = 22.5 nM T73482 CPZ89B 135314564 Ki = 8.14 nM T73482 C75NWT 136227358 IC50 > 30000 nM T73482 C9WUL6 137632260 Ki = 14 nM T73482 C24MIN 137632538 IC50 > 10000 nM T73482 C61SQF 137633141 Ki = 2.44 nM T73482 C3UBF8 137634720 IC50 = 489 nM T73482 CH4KC1 137635768 Ki = 42.3 nM T73482 C0BRG6 137636340 IC50 = 113 nM T73482 C0G8TB 137637342 IC50 = 3239 nM T73482 C4W3YF 137637374 Ki = 8.99 nM T73482 C7FUO1 137638475 Ki = 31.6 nM T73482 C04EGF 137638805 IC50 = 293 nM T73482 CYB93R 137638895 IC50 = 5020 nM T73482 CZ91SV 137638898 IC50 > 10000 nM T73482 CQ5J0X 137639504 Ki = 320 nM T73482 CT90FM 137640166 IC50 > 10000 nM T73482 C79OCZ 137641214 Ki = 7.25 nM T73482 CIPJ41 137641369 IC50 = 1963 nM T73482 C5OXI1 137642484 IC50 = 759 nM T73482 CX3MK7 137642825 IC50 = 1895 nM T73482 CNM4F9 137643075 Ki = 541 nM T73482 C2DIV4 137644135 IC50 = 1910 nM T73482 C6M0BL 137644509 IC50 = 216 nM T73482 C9ABK7 137644534 IC50 = 327 nM T73482 C6KM9A 137645155 Ki = 6.37 nM T73482 C2MRK0 137645329 Ki = 18.9 nM T73482 C9GP2E 137645716 Ki = 10 nM T73482 CC6KI7 137646689 IC50 = 3918 nM T73482 CF98UE 137647371 IC50 = 502 nM T73482 C2BQ4U 137648163 IC50 = 1010 nM T73482 C4VD0P 137649196 IC50 > 10000 nM T73482 CLZ2N8 137649834 IC50 = 226 nM T73482 C1TW0K 137650367 Ki = 12 nM T73482 C7X0SU 137651169 Ki = 849 nM T73482 CR5F0I 137652411 IC50 = 303 nM T73482 C36YGM 137653736 Ki = 389 nM T73482 CPE53S 137654752 Ki = 1.92 nM T73482 C08XSJ 137655492 IC50 > 10000 nM T73482 C1MJG9 137655850 IC50 = 1636 nM T73482 C7R3IU 137656102 Ki = 14 nM T73482 CQ0UG7 137657078 IC50 = 2973 nM T73482 C7VFU4 137657849 IC50 = 736 nM T73482 CF7Q6D 137658206 IC50 = 908 nM T73482 C63RQO 137658775 IC50 = 517 nM T73482 C89FIO 137659457 IC50 = 1776 nM T73482 CNH3U0 137660075 IC50 > 10000 nM T73482 C38LZW 137660448 Ki = 11.2 nM T73482 CQ0J2X 137660887 IC50 = 401 nM T73482 CUMN86 137662108 Ki = 66 nM T73482 CNX2Q5 137662177 Ki = 12.9 nM T73482 CZ4S3O 144671360 IC50 = 89 nM T73482 CF0Z8D 145714283 Ki = 15.85 nM T73482 CS9B7W 145971593 Ki = 1.97 nM T73482 C27YQH 145975735 Ki = 187 nM T73482 C7CO2P 145977763 Ki = 17.8 nM T73482 C6VWK3 145979924 Ki = 4800 nM T73482 CGRU50 145989367 Ki = 5400 nM T73482 C3M1WQ 145994245 Ki = 3100 nM T73482 CQD73L 155515631 Ki = 502 nM T73482 C2B1ZG 155517489 Ki > 10 nM T73482 CH3MT0 155519961 Ki > 10 nM T73482 C9D3AS 155520434 Ki = 5.89 nM T73482 CF1N4P 155524300 Ki = 461 nM T73482 CWL04C 155524427 Ki = 4.34 nM T73482 CB3JY5 155525887 Ki = 5.51 nM T73482 C5EM4D 155532688 Ki = 9.35 nM T73482 C4VQ8A 155543013 Ki > 10 nM T73482 CP7I4W 155543165 Ki > 10 nM T73482 CFMK42 155543728 Ki = 101 nM T73482 CIY9N3 155554119 Ki > 10 nM T73482 CQ30PW 155557825 Ki = 20.9 nM T73482 CRDS43 155566853 Ki = 842 nM T73482 CM93SV 155567436 Ki = 7.45 nM T73482 CQ1RW5 155568320 Ki > 10000 nM T73482 D01SUL 9869934 Ki = 5.012 nM T73482 D02MDC 9981404 Ki = 900 nM T73482 D08MXD 73349109 Ki = 1.1 nM T73482 D0J3PJ 4331799 Ki = 22 nM T73482 D0KP3K 10065953 Ki = 8.7 nM T73482 D0R4BT 10046856 Ki = 100 nM T73482 D0U0TS 10408514 IC50 > 10000 nM T73482 D0UZ4J 6604926 Ki = 14 nM T36483 D0VA0I 10077130 IC50 = 1.1 nM T36483 D0PU8T 10459564 IC50 = 31.62 nM T36483 D08ELM 9832212 IC50 = 5 nM T36483 CO6X0U 128205 IC50 = 9000 nM T36483 C98PBF 752812 IC50 = 10000 nM T36483 CX79RF 807100 IC50 = 1120 nM T36483 C0DXY9 877874 IC50 = 1680 nM T36483 C1HPL9 1047175 IC50 = 900 nM T36483 C4U2DR 1047178 IC50 = 2866 nM T36483 C82PVQ 1047179 IC50 = 98 nM T36483 CWTG42 1048267 IC50 = 199.53 nM T36483 C48FJQ 1361448 IC50 = 3120 nM T36483 CYN6E5 2858257 IC50 = 33 nM T36483 CCIE45 2858875 IC50 = 65 nM T36483 C1QC2W 3109060 IC50 = 316.23 nM T36483 CLBW26 3378161 IC50 = 1410 nM T36483 CXU4P3 3751851 IC50 = 359 nM T36483 CZS63L 4259181 IC50 = 56 nM T36483 C8LYU1 4314709 IC50 = 964 nM T36483 CD4YR5 7006478 EC50 > 800000 nM T36483 C2ST5A 9801767 IC50 = 700 nM T36483 CO28KU 9805672 IC50 = 1000 nM T36483 CB6E8G 9808447 EC50 = 760 nM T36483 CSV54F 9809471 EC50 = 1000 nM T36483 C8UDN9 9810474 IC50 = 1600 nM T36483 CVDI10 9810475 IC50 = 6700 nM T36483 CK1NW8 9810477 EC50 = 2900 nM T36483 C3B7WM 9825804 IC50 = 20 nM T36483 CZWL57 9831601 IC50 = 30000 nM T36483 C2HY1Z 9831828 IC50 = 5000 nM T36483 C6CRK1 9831948 IC50 = 5600 nM T36483 CAW29Z 9844209 IC50 = 22 nM T36483 C69RDJ 9847494 IC50 = 150 nM T36483 CBKT76 9851501 EC50 = 1200 nM T36483 C75JUE 9853816 IC50 = 270 nM T36483 CSB56V 9855084 EC50 = 8000 nM T36483 CN48IZ 9865055 IC50 = 27 nM T36483 CR80DB 9869359 IC50 = 21.5 nM T36483 CGET90 9875040 EC50 = 21000 nM T36483 CWI9F8 9875337 EC50 = 1100 nM T36483 CW18TC 9886874 IC50 = 15 nM T36483 CC85QB 9889179 IC50 = 10 nM T36483 CRK15D 9890926 Ki = 11 nM T36483 CXWF97 9895920 EC50 = 460 nM T36483 CV8GN6 9896668 IC50 > 100000 nM T36483 CO93LE 9897054 IC50 = 25 nM T36483 C8H1QX 9908345 IC50 = 22 nM T36483 CG36KH 9919038 IC50 = 570 nM T36483 CC75WO 9931987 IC50 = 10 nM T36483 CT67FC 9934461 IC50 = 23 nM T36483 C7NWE2 9937578 EC50 = 3900 nM T36483 CL28YV 9951647 IC50 = 6.3 nM T36483 CJH61W 9960837 EC50 = 1000 nM T36483 CB7PQ1 9961058 EC50 = 510 nM T36483 CC3BO7 9962227 EC50 = 1000 nM T36483 CBI45Z 9982475 EC50 = 185000 nM T36483 CK0OF1 9986700 EC50 = 800000 nM T36483 CYH1Z5 9986822 EC50 = 400 nM T36483 CXIF90 9987318 EC50 = 600000 nM T36483 CAHV37 10000177 IC50 = 52 nM T36483 CEOA76 10010285 EC50 = 200 nM T36483 C6RMX0 10032001 EC50 = 109300 nM T36483 CWZ42G 10032227 EC50 = 700 nM T36483 C0UD8L 10054163 EC50 = 15000 nM T36483 C2UJ7B 10054787 EC50 = 730000 nM T36483 CJ9P1Z 10078162 EC50 = 19000 nM T36483 C60PZS 10078455 EC50 > 1200000 nM T36483 C03XAC 10079418 EC50 = 10 nM T36483 C82XUE 10095734 IC50 = 20 nM T36483 CU25DY 10099272 EC50 > 800000 nM T36483 C19QPS 10101423 EC50 = 270 nM T36483 C8K9OD 10120960 IC50 = 1200 nM T36483 C1TB4S 10161572 IC50 = 350 nM T36483 CO5NT2 10162707 IC50 = 830 nM T36483 CN0ZW5 10164471 IC50 = 4440 nM T36483 C7XNK5 10184176 IC50 = 1100 nM T36483 CT96NH 10204371 IC50 = 6600 nM T36483 CG52LT 10206026 IC50 = 430 nM T36483 CB32WA 10227544 IC50 = 2100 nM T36483 CBSL17 10246587 Ki = 12 nM T36483 CNG2M1 10257805 EC50 = 200000 nM T36483 CUO92S 10259068 EC50 = 500 nM T36483 C19IWT 10260648 EC50 > 800000 nM T36483 CMX30H 10276545 IC50 = 130 nM T36483 CLE90J 10278388 IC50 = 3700 nM T36483 CT69SW 10279248 IC50 = 3200 nM T36483 C28CZY 10300275 IC50 = 120 nM T36483 CME8H2 10325208 EC50 = 70000 nM T36483 CD7B9J 10328351 IC50 = 3100 nM T36483 CF9Q3K 10345602 Ki = 1900 nM T36483 CKZ0T7 10348644 EC50 = 1200 nM T36483 CSU8H4 10350578 EC50 = 500 nM T36483 CCGH96 10350886 IC50 = 7.5 nM T36483 CL9EB4 10351173 EC50 = 3300 nM T36483 C4AZW0 10371218 EC50 = 1300 nM T36483 C8EPN7 10390481 Ki = 6600 nM T36483 CB65WG 10394462 EC50 > 800000 nM T36483 COZ92M 10415062 EC50 > 800000 nM T36483 CM3ZX0 10416585 EC50 = 415000 nM T36483 C4QX8B 10416597 EC50 = 235000 nM T36483 CI5AZ6 10416607 EC50 = 800000 nM T36483 CO8U9A 10416608 EC50 > 800000 nM T36483 C0C3ZK 10416646 EC50 = 200 nM T36483 CGDA78 10416780 EC50 = 350000 nM T36483 C1Q6JH 10417097 EC50 = 140 nM T36483 C6KA0H 10418424 EC50 = 24500 nM T36483 CHAN91 10439025 EC50 > 800000 nM T36483 C21MID 10439062 EC50 = 500000 nM T36483 C8M7SV 10441247 EC50 > 800000 nM T36483 CXZJ53 10461499 EC50 = 11700 nM T36483 C02WYD 10461589 EC50 = 28000 nM T36483 CTY5H0 10462502 EC50 = 400000 nM T36483 CO02ET 10484360 EC50 = 21400 nM T36483 CE0PF1 10484500 EC50 > 800000 nM T36483 C4VN0A 10526120 IC50 = 80 nM T36483 CMVI23 10557086 IC50 = 24 nM T36483 CRFI52 10622095 IC50 = 90 nM T36483 C2FLV0 10628873 IC50 = 29 nM T36483 CTF43Q 10741717 IC50 = 80 nM T36483 CI96NX 10747898 EC50 = 1800 nM T36483 CF9Y3J 10771636 IC50 = 19 nM T36483 C4SQ5G 10818136 EC50 = 720 nM T36483 CIR3E1 10819322 IC50 = 300 nM T36483 CQ6G0B 10925413 IC50 = 1500 nM T36483 CD25QZ 11502485 IC50 = 25 nM T36483 C5ZWX6 11502697 IC50 = 1000 nM T36483 CNOC42 11503433 IC50 = 46 nM T36483 CQE03H 11508687 IC50 = 850 nM T36483 CRT82D 11509594 IC50 = 325 nM T36483 CA7D8B 11515660 IC50 = 1500 nM T36483 C43BGM 11516923 IC50 = 900 nM T36483 CVT96B 11537143 IC50 = 300 nM T36483 C2BM8L 11544606 IC50 = 150 nM T36483 CR6UX2 11544845 IC50 = 210 nM T36483 C4M3HK 11553497 IC50 = 11 nM T36483 CQZI28 11559190 IC50 = 1250 nM T36483 C8RZJ4 11567556 IC50 = 14 nM T36483 C38CUB 11576348 IC50 = 100 nM T36483 C9PG8E 11582568 IC50 = 26 nM T36483 C1TE7Q 11583548 IC50 = 25 nM T36483 C9QN7H 11603083 IC50 = 143 nM T36483 CO2P9S 11610042 IC50 = 250 nM T36483 C5B9MN 11611061 IC50 = 13 nM T36483 CN5C2X 11611425 IC50 = 204 nM T36483 CN9VJ8 11618945 IC50 = 29 nM T36483 C3H2TL 11624004 IC50 > 5000 nM T36483 C23DJQ 11639231 IC50 = 550 nM T36483 CAT1C0 11645276 IC50 = 4000 nM T36483 CO37QK 11647382 IC50 = 19 nM T36483 C4CY7V 11652756 IC50 = 1100 nM T36483 CI6QM8 11661666 IC50 = 28 nM T36483 CD5SX3 11674764 IC50 = 725 nM T36483 C6UGL9 11682882 IC50 = 467 nM T36483 CO92VG 11684648 IC50 = 50 nM T36483 CS7FH4 11688420 IC50 = 2100 nM T36483 CV4OW8 11690507 IC50 = 19 nM T36483 C6VQH5 11691128 IC50 = 44 nM T36483 C4AYW2 11697104 IC50 = 35 nM T36483 CD2M6O 11702885 IC50 = 325 nM T36483 CPJG59 11703925 IC50 = 3500 nM T36483 CIYF09 11712191 IC50 > 300 nM T36483 C8G1ZT 11718309 IC50 = 3681 nM T36483 CV9Q1B 11758525 EC50 = 800 nM T36483 C9K6JA 11764645 EC50 > 800000 nM T36483 C4JG1W 11803290 IC50 = 25 nM T36483 CZ74PR 11803426 EC50 = 3700 nM T36483 CLDX73 11803455 IC50 = 193000 nM T36483 CDXL23 11818750 EC50 = 2000 nM T36483 C90MCQ 12018757 IC50 = 2990 nM T36483 CG6Q4B 12018758 IC50 = 910 nM T36483 CP15ZG 12018759 IC50 = 990 nM T36483 CT7Z2V 12018762 IC50 = 140 nM T36483 C2B8GR 15887956 IC50 = 4000 nM T36483 CKPY93 15887958 IC50 = 65000 nM T36483 C8QO3Z 15887960 IC50 = 40000 nM T36483 CKVM71 16046150 IC50 = 18 nM T36483 CG2NT3 16100342 IC50 = 41 nM T36483 CCG1W9 16100343 IC50 = 845 nM T36483 CY5FP4 16100350 IC50 = 37 nM T36483 CRF9T3 16100351 IC50 = 53 nM T36483 CRNU53 16100352 IC50 = 28 nM T36483 CQD1R6 16100353 IC50 = 481 nM T36483 CM07ZP 17187522 IC50 = 770 nM T36483 CPW18A 17187534 IC50 = 1100 nM T36483 CPFW98 17187609 IC50 = 970 nM T36483 CZWL06 17222599 IC50 = 199.53 nM T36483 C3Y2KE 17222608 IC50 = 1800 nM T36483 CHVR74 22611774 IC50 = 28000 nM T36483 CVM5Q1 22611776 IC50 > 10000 nM T36483 C5LH4U 22611792 IC50 = 2000 nM T36483 C2WR9E 22611889 IC50 > 10000 nM T36483 C4V7BI 22645287 IC50 = 8000 nM T36483 C7EQ5O 23628249 IC50 = 7.6 nM T36483 C5EG4O 23630913 IC50 = 22 nM T36483 CN1EW7 23630914 IC50 = 200 nM T36483 CE86TG 23630915 IC50 = 80 nM T36483 C1PKN9 23631103 IC50 = 17 nM T36483 C69YXL 23631104 IC50 = 26 nM T36483 CD7WU0 23631105 IC50 = 25 nM T36483 CSC80P 23631106 IC50 = 26 nM T36483 C4C5JA 23631184 IC50 = 19 nM T36483 CS89QV 23631185 IC50 = 13 nM T36483 C26ENM 23631186 IC50 = 21 nM T36483 CSKH79 23631187 IC50 = 11 nM T36483 C83UCD 23631188 IC50 = 8 nM T36483 CO5CD4 23631275 IC50 = 33.5 nM T36483 CNGH14 23631277 IC50 = 762 nM T36483 CM93CL 23631278 IC50 = 550 nM T36483 CI8HF9 23631279 IC50 = 37.5 nM T36483 C2F6CI 23631374 IC50 = 15.5 nM T36483 CZR10M 23631375 IC50 = 1101 nM T36483 CHN4X8 23631376 IC50 = 18.5 nM T36483 CEP5C7 23631377 IC50 = 101 nM T36483 CD4MH1 23631464 IC50 = 25 nM T36483 C6RH3X 23631554 IC50 = 224 nM T36483 CXUF30 23631639 IC50 = 153 nM T36483 C4L9ZI 23631640 IC50 = 295 nM T36483 CEI32D 23631809 IC50 = 600 nM T36483 CH9AO6 23631810 IC50 = 113 nM T36483 CH25IR 23631811 IC50 = 8 nM T36483 C59OSL 23631812 IC50 = 15 nM T36483 C9GVK3 23631813 IC50 = 16.5 nM T36483 CNB2Z0 23631900 IC50 = 600 nM T36483 CP23YQ 24830436 Ki = 17 nM T36483 CC65LO 24830595 Ki = 6.1 nM T36483 CO8MA9 24878827 Ki = 13 nM T36483 C6IX1G 24878828 Ki = 20 nM T36483 C0N4AJ 24878829 Ki = 30 nM T36483 C6W9PK 24878871 Ki = 6.4 nM T36483 CC2E7B 24878872 Ki = 6.5 nM T36483 CQ4VO9 24878873 Ki = 6.2 nM T36483 C1DJS3 24878874 Ki = 4.4 nM T36483 C45EUD 24878875 Ki = 4.8 nM T36483 CB6P4R 24878927 Ki = 11 nM T36483 CV7SN0 24878928 Ki = 10 nM T36483 CDX49C 24878929 Ki = 44 nM T36483 CBCR43 24878930 Ki = 4.1 nM T36483 CJB97D 24878981 Ki = 89 nM T36483 C6Y5DM 24878982 Ki = 3.7 nM T36483 CCV09N 24878983 Ki = 5.9 nM T36483 CAF0C7 24878984 Ki = 11 nM T36483 CC4A6K 24879035 Ki = 367 nM T36483 CMH5P1 24879036 Ki = 1.8 nM T36483 CBE9L3 24879037 Ki = 11 nM T36483 C1MXQ6 24879038 Ki = 5.9 nM T36483 CFU61L 24879079 Ki = 11 nM T36483 C9RND0 44264660 Ki = 14000 nM T36483 CQ2R6H 44280522 IC50 = 7600 nM T36483 CE9G2Z 44280585 EC50 = 760 nM T36483 CK18FO 44280607 EC50 = 28000 nM T36483 CBKV73 44280608 EC50 = 1700 nM T36483 CN95GQ 44280649 IC50 = 4000 nM T36483 CQ95NM 44280650 IC50 = 1400 nM T36483 CFZX80 44280651 EC50 = 5000 nM T36483 CK34GX 44280660 IC50 = 3000 nM T36483 CY8WM5 44280667 EC50 = 5800 nM T36483 CCF1H9 44280683 EC50 = 8000 nM T36483 C0PFB8 44280685 EC50 = 1300 nM T36483 CYV23Q 44280703 IC50 = 7000 nM T36483 CZBU08 44280731 IC50 = 10000 nM T36483 C47GQL 44280767 EC50 = 1000 nM T36483 CE9LF7 44280768 EC50 = 3100 nM T36483 CHP49J 44280804 EC50 = 2000 nM T36483 CU0K5H 44280805 IC50 = 25000 nM T36483 C78GZV 44280822 EC50 = 4200 nM T36483 CK8W4F 44280835 IC50 = 27000 nM T36483 CFW53T 44280876 IC50 = 10000 nM T36483 C4SZK0 44280877 EC50 = 2100 nM T36483 C9T8SX 44280878 IC50 = 46000 nM T36483 CXAT87 44280898 IC50 = 10000 nM T36483 CCS25K 44280899 IC50 = 4400 nM T36483 C9C0HI 44280905 IC50 = 2600 nM T36483 C2JD9S 44280935 EC50 = 2400 nM T36483 CG7X6F 44280936 EC50 = 7900 nM T36483 C84DSX 44280949 EC50 = 1200 nM T36483 CC6HB0 44280954 IC50 = 16000 nM T36483 CS5FV7 44280955 EC50 = 4900 nM T36483 CJMQ02 44281047 EC50 = 14000 nM T36483 C18ZQK 44281069 IC50 = 13000 nM T36483 C0GKP4 44281070 IC50 = 2300 nM T36483 C3QA2W 44281079 IC50 = 2400 nM T36483 CT27UM 44281080 IC50 = 2900 nM T36483 CDH74W 44281081 IC50 = 2000 nM T36483 C6J3CG 44281172 EC50 = 10500 nM T36483 CM29OK 44281173 IC50 = 9000 nM T36483 C7C4ZT 44281174 IC50 = 18000 nM T36483 CV2Q5K 44281237 EC50 = 2600 nM T36483 C2EU9P 44281263 IC50 = 5000 nM T36483 C50SCD 44281264 IC50 = 56000 nM T36483 CW94SR 44281289 EC50 = 9700 nM T36483 C5P7QN 44289942 IC50 > 100000 nM T36483 CF4J5T 44289951 IC50 > 100000 nM T36483 CQ32XB 44289954 IC50 = 8000 nM T36483 CPI04Z 44290058 IC50 = 5400 nM T36483 C51LBS 44290059 IC50 = 6200 nM T36483 C0LT9V 44290102 IC50 = 2700 nM T36483 CYDK89 44290104 IC50 = 10000 nM T36483 CLPO09 44290110 IC50 = 60000 nM T36483 C8LZ7F 44290166 IC50 = 4100 nM T36483 CHI87Y 44290181 IC50 = 5000 nM T36483 C2R4LT 44290206 IC50 = 24000 nM T36483 CYS73M 44290207 IC50 = 24000 nM T36483 CRP2J4 44290231 IC50 = 5700 nM T36483 CGT83M 44290234 IC50 = 8200 nM T36483 C7TF4J 44290251 IC50 = 94000 nM T36483 CWM53Q 44290276 IC50 = 53000 nM T36483 C2PY9U 44290300 IC50 = 2700 nM T36483 C74XUM 44305776 IC50 = 300 nM T36483 CGF8T4 44305882 IC50 = 1250 nM T36483 CEA1W6 44305896 IC50 = 870 nM T36483 C8D0JY 44305897 IC50 = 524 nM T36483 C9OL6V 44305939 IC50 = 4500 nM T36483 CH1ZU6 44305942 IC50 = 1750 nM T36483 CN0BF5 44305944 IC50 = 3200 nM T36483 CY7D3U 44305948 IC50 = 100 nM T36483 CZL50Q 44305953 IC50 = 4900 nM T36483 C2IQS3 44305954 IC50 = 100 nM T36483 C0EM9F 44305955 IC50 = 9600 nM T36483 CB90FJ 44306065 IC50 = 1230 nM T36483 CNR6Y4 44306066 IC50 = 2625 nM T36483 C7AC4M 44306076 IC50 = 6875 nM T36483 CUG1B0 44306336 IC50 = 600 nM T36483 CGX38W 44306402 IC50 = 310 nM T36483 CRIA53 44306403 IC50 = 230 nM T36483 C5QFP0 44306404 IC50 = 1000 nM T36483 C4IXK0 44306499 IC50 = 1300 nM T36483 CO70XF 44306500 IC50 = 140 nM T36483 CT2JH0 44306501 IC50 = 70 nM T36483 CDV41R 44306540 IC50 = 640 nM T36483 C2FYC6 44306599 IC50 = 100 nM T36483 C9QYF1 44306611 IC50 = 400 nM T36483 CFEN89 44306612 IC50 = 36500 nM T36483 C9C6OD 44306657 IC50 = 4800 nM T36483 CT7L9J 44306658 IC50 = 3500 nM T36483 CAVY39 44306659 IC50 = 400 nM T36483 C0QVF7 44306660 IC50 = 900 nM T36483 CW6R7A 44306696 IC50 = 2000 nM T36483 C1G9RQ 44306697 IC50 = 240 nM T36483 CY9QL2 44306698 IC50 = 200 nM T36483 CM90EW 44306708 IC50 = 1300 nM T36483 C8VJ7B 44306732 IC50 = 500 nM T36483 CR9J2L 44306761 IC50 = 440 nM T36483 CT58LC 44306762 IC50 = 100 nM T36483 CJL6R7 44306894 IC50 = 900 nM T36483 C20CMS 44306903 IC50 = 2300 nM T36483 CRV4M7 44309450 IC50 = 2000 nM T36483 CE85SQ 44309461 IC50 = 230 nM T36483 CB20GZ 44309471 IC50 = 70 nM T36483 C9RP0K 44309472 IC50 = 500 nM T36483 CQJD59 44309477 IC50 = 120 nM T36483 C81MZX 44309730 IC50 = 480 nM T36483 CU4TG6 44309750 IC50 = 160 nM T36483 CID42J 44309751 IC50 = 330 nM T36483 C7Y1QM 44309776 IC50 = 430 nM T36483 C9SBO3 44309777 IC50 = 310 nM T36483 CF98YJ 44309838 IC50 = 22000 nM T36483 CJU6I8 44309958 IC50 = 35 nM T36483 CLFB39 44309959 IC50 = 70 nM T36483 C7MVQ9 44310191 IC50 = 90 nM T36483 CW2Z1T 44310308 IC50 = 60 nM T36483 C1ZCH0 44310323 IC50 = 130 nM T36483 CJN6H3 44315779 IC50 > 10000 nM T36483 C8LQ3E 44315780 IC50 = 20000 nM T36483 C5XE1O 44315792 IC50 = 5000 nM T36483 CPT6R4 44315793 IC50 = 7000 nM T36483 C2TE0B 44316045 IC50 = 2000 nM T36483 C7P1CL 44316059 IC50 = 7000 nM T36483 CDVZ48 44316106 IC50 = 4000 nM T36483 C9B8CD 44316156 IC50 = 800 nM T36483 CUBM67 44316184 IC50 = 1000 nM T36483 CAI6P7 44316522 IC50 = 300 nM T36483 C8DRY2 44316532 IC50 = 3000 nM T36483 CYTL98 44316560 IC50 = 11000 nM T36483 C6QU9I 44316563 IC50 > 50000 nM T36483 C2D5ZR 44324193 IC50 = 700 nM T36483 CIJF13 44328197 IC50 = 9000 nM T36483 CKC07Y 44328340 IC50 = 3100 nM T36483 C7M8TH 44328342 IC50 = 13000 nM T36483 C1SG3Y 44328381 IC50 = 3400 nM T36483 C5HI4J 44328383 IC50 = 9700 nM T36483 CL2FU7 44328523 IC50 = 300 nM T36483 CNS8K1 44328562 IC50 = 6000 nM T36483 C3B6RN 44328579 IC50 = 1324 nM T36483 CV5XZ1 44328647 IC50 = 734 nM T36483 C8I3EG 44328728 IC50 = 1500 nM T36483 CWI9D5 44338787 IC50 = 500 nM T36483 CM05QN 44338791 IC50 = 90 nM T36483 C5A6JX 44338864 IC50 = 360 nM T36483 C89OIS 44338865 IC50 = 5000 nM T36483 CQ6I8E 44338875 IC50 = 500 nM T36483 C73QCH 44338882 IC50 = 600 nM T36483 CLUN47 44338885 IC50 = 1600 nM T36483 CHY5J0 44338886 IC50 = 3300 nM T36483 CVA3B2 44338887 IC50 > 10000 nM T36483 CCLA27 44338895 IC50 = 2000 nM T36483 C3V2YS 44338903 IC50 > 10000 nM T36483 CZ69BK 44338917 IC50 = 1000 nM T36483 C20HJG 44338928 IC50 > 10000 nM T36483 C91WXN 44338929 IC50 = 130 nM T36483 CI1Q0K 44338944 IC50 = 70 nM T36483 CM8C9F 44338946 IC50 = 400 nM T36483 CMKH71 44339001 IC50 = 2210 nM T36483 C9ZK0U 44339002 IC50 = 290 nM T36483 CY5V7Z 44339029 IC50 = 120 nM T36483 C2AE6H 44339030 IC50 = 6420 nM T36483 CWRP93 44339048 IC50 > 10000 nM T36483 CIE4V2 44339055 IC50 = 3220 nM T36483 CD3O4Z 44339056 IC50 = 5000 nM T36483 CUP92F 44339060 IC50 = 12000 nM T36483 CO45AF 44339061 IC50 > 40000 nM T36483 CG4R7X 44339070 IC50 = 500 nM T36483 CSY5W6 44339157 IC50 = 1310 nM T36483 C3BM0F 44339173 IC50 = 130 nM T36483 C0W4UH 44354022 EC50 = 31000 nM T36483 CZ3P4T 44354052 EC50 = 800000 nM T36483 C4AFJ8 44354055 EC50 = 10 nM T36483 CB3Y0N 44354062 EC50 > 800000 nM T36483 C2IA5K 44354106 EC50 = 120 nM T36483 CX1B6H 44354107 EC50 = 40000 nM T36483 CC1H6G 44354108 EC50 = 130 nM T36483 C4C8FX 44354285 EC50 = 150 nM T36483 C2MVY1 44354323 EC50 = 30 nM T36483 C84VLR 44354387 EC50 = 600000 nM T36483 C4BY2H 44354460 EC50 = 260000 nM T36483 CL94CB 44403839 IC50 = 400 nM T36483 CGN3M7 44408615 IC50 = 730 nM T36483 CV14NJ 44408616 IC50 = 150 nM T36483 C48NRV 44408709 IC50 = 700 nM T36483 CV2FB8 44408711 IC50 = 390 nM T36483 CL8ET4 44408851 IC50 = 60 nM T36483 CGZ5L1 44408873 IC50 = 15 nM T36483 CPHR30 44408874 IC50 = 155 nM T36483 CJ1WK6 44409029 IC50 = 500 nM T36483 C10MZB 44409033 IC50 = 300 nM T36483 CWLA42 44409034 IC50 = 28 nM T36483 C5BN2E 44409039 IC50 = 2151 nM T36483 CFGH09 44409050 IC50 = 800 nM T36483 C8WJN0 44409057 IC50 = 25 nM T36483 C85SAC 44409062 IC50 = 500 nM T36483 C2ME6W 44409074 IC50 = 50 nM T36483 C7IBZ8 44409076 IC50 = 300 nM T36483 CO85YX 44409077 IC50 = 219 nM T36483 C3I2XK 44409082 IC50 = 125 nM T36483 CQ9ZP8 44409083 IC50 = 1250 nM T36483 C0AM4W 44409228 IC50 = 275 nM T36483 CCL1W8 44409232 IC50 = 30 nM T36483 CFI18T 44409248 IC50 = 50 nM T36483 CPM0H5 44409253 IC50 = 100 nM T36483 C49FKT 44409259 IC50 = 68 nM T36483 CK82DA 44409265 IC50 = 1000 nM T36483 C3E8ZK 44409278 IC50 = 290 nM T36483 C14SBI 44409289 IC50 = 800 nM T36483 C9V7SR 44416466 IC50 = 426 nM T36483 CGU2I4 44416487 IC50 = 7000 nM T36483 CT5AF6 44416541 IC50 = 1500 nM T36483 CAC6W5 44416542 IC50 = 200 nM T36483 CXO31W 44416562 IC50 = 150 nM T36483 CVQ20M 44416563 IC50 = 3500 nM T36483 CJB97L 44416567 IC50 = 623 nM T36483 CVD1L4 44416588 IC50 = 2000 nM T36483 CIEH73 44416634 IC50 = 7000 nM T36483 C16OSE 44416654 IC50 = 217 nM T36483 CB6K0L 44416672 IC50 = 8000 nM T36483 CIK31H 44416690 IC50 = 150 nM T36483 C2WUH0 44416691 IC50 = 62 nM T36483 C0DPY7 44416717 IC50 = 3750 nM T36483 CBD0K2 44416724 IC50 = 5000 nM T36483 CO40PE 44416740 IC50 = 74 nM T36483 CN3IR6 44418837 IC50 = 80 nM T36483 C73PLG 44418838 IC50 = 28 nM T36483 CIR8G5 44418839 IC50 = 72 nM T36483 CEV27S 44418840 IC50 = 829 nM T36483 C8G3KX 44418842 IC50 = 38.5 nM T36483 CD51EF 44418844 IC50 = 147 nM T36483 CH43LA 44418846 IC50 = 70 nM T36483 C3VI2T 44418847 IC50 = 1374 nM T36483 CF0KU1 44418848 IC50 = 97 nM T36483 C8H0DE 44418849 IC50 = 16.5 nM T36483 CBZ93Y 44418850 IC50 = 15 nM T36483 C9DOX5 44418854 IC50 = 28 nM T36483 COX93N 44418855 IC50 = 12 nM T36483 C5NRG9 44418858 IC50 = 11 nM T36483 CEH4F5 44428104 Ki = 4.3 nM T36483 CR2ZA7 44432691 IC50 = 3600 nM T36483 CPY1T2 44432692 IC50 = 350 nM T36483 CG8V5A 44432693 IC50 = 43 nM T36483 CR6PH9 44432704 IC50 = 130 nM T36483 CPCF39 44432705 IC50 = 285 nM T36483 CW51XH 44432706 IC50 = 263 nM T36483 CRT4L1 44432707 IC50 = 115 nM T36483 CPOM02 44432708 IC50 = 29 nM T36483 CG0Q7L 44432710 IC50 = 3300 nM T36483 CQK89F 44432711 IC50 = 12 nM T36483 C7KMN5 44432712 IC50 = 16 nM T36483 C1RVW9 44432713 IC50 = 36 nM T36483 CV5Z8K 44432714 IC50 = 11 nM T36483 C6VPH0 44432715 IC50 = 47 nM T36483 C70NXO 44432716 IC50 = 1320 nM T36483 CO9IN1 44432717 IC50 = 145 nM T36483 C9FB6J 44432718 IC50 = 22 nM T36483 COP92K 44432719 IC50 = 2144 nM T36483 C2N4DU 44432720 IC50 = 207 nM T36483 C42LFE 44432721 IC50 = 88 nM T36483 C6LU8S 44432756 IC50 = 440 nM T36483 CL1ON3 44432763 IC50 = 65 nM T36483 CG35DW 44432767 IC50 = 31.5 nM T36483 CFD86M 44432770 IC50 = 137.5 nM T36483 CQU32G 44432771 IC50 = 225 nM T36483 CMDL57 44432772 IC50 = 46.5 nM T36483 C5EK6H 44432773 IC50 = 10 nM T36483 C8E9BN 44432774 IC50 = 120 nM T36483 CPR7M9 44432775 IC50 = 29 nM T36483 CDV3F2 44432778 IC50 = 328 nM T36483 C8T3YF 44432779 IC50 = 13 nM T36483 C20FMS 44432783 IC50 = 15.5 nM T36483 CZS35O 44432786 IC50 = 330 nM T36483 C7PE6B 44432790 IC50 = 10 nM T36483 CC1V7G 44432791 IC50 = 20.5 nM T36483 CWHP50 44432795 IC50 = 63.5 nM T36483 CU36DS 44432798 IC50 = 14.5 nM T36483 C7XSD8 44432803 IC50 = 7 nM T36483 C2M6BU 44432806 IC50 = 85.5 nM T36483 CXZ5V1 44432814 IC50 = 7.5 nM T36483 C5QCT4 44432817 IC50 = 14.5 nM T36483 C8Y1ER 44432831 IC50 = 12000 nM T36483 C6MW3X 44432833 IC50 = 580 nM T36483 CL3E7S 44432836 IC50 = 90 nM T36483 CO0NA4 44432839 IC50 = 9170 nM T36483 C1RU9S 44432840 IC50 = 3139 nM T36483 C4N9BO 44432842 IC50 = 225 nM T36483 C4GPB7 44432843 IC50 = 12.5 nM T36483 C0PO8C 44584151 IC50 = 20000 nM T36483 C3ZGS2 44826171 EC50 = 1900 nM T36483 CE5Q1R 44826172 EC50 = 1900 nM T36483 CDXT67 49766539 IC50 = 520 nM T36483 C4AZ6G 49766546 IC50 = 2200 nM T36483 C1ER8F 50910530 IC50 = 3000 nM T36483 C3U5JP 50910534 IC50 = 520 nM T36483 CX5K9E 50910535 IC50 = 710 nM T36483 C29DEG 50910547 IC50 = 1290 nM T36483 CPYE39 50910548 IC50 = 3160 nM T36483 CE03PW 50910549 IC50 = 2640 nM T36483 C8N0ID 51003683 IC50 = 340 nM T36483 C0JNG8 52940892 Ki = 144 nM T36483 C35CDM 52940897 Ki = 337 nM T36483 C3FX0H 52942074 Ki = 240 nM T36483 CA42IG 52942093 Ki = 42 nM T36483 C9SET2 52946929 Ki = 250 nM T36483 CBC61R 52946957 Ki = 49 nM T36483 C3H4PS 52947767 Ki = 12 nM T36483 C8AQ3X 52948306 Ki = 75 nM T36483 C5EO4F 52949425 Ki = 61 nM T36483 CBJ6D3 52949514 Ki = 15 nM T36483 CVBF92 53245432 IC50 = 600 nM T36483 CH05IO 53245434 IC50 = 480 nM T36483 CUG2I9 53245435 IC50 = 390 nM T36483 C9AD3Q 53245451 IC50 = 380 nM T36483 C4G2IS 53245483 IC50 = 2280 nM T36483 CNJL95 56668146 IC50 > 100000 nM T36483 C7C6XG 56671606 IC50 = 3900 nM T36483 CQN67G 56949066 IC50 = 970 nM T36483 C8JZM0 57404483 IC50 = 8.1 nM T36483 CL08XW 57404484 IC50 = 4.6 nM T36483 C72MWG 57404504 IC50 = 6.4 nM T36483 C6I9BF 57892463 IC50 = 31.62 nM T36483 CN9C2H 58187662 Ki = 35 nM T36483 C5UYB6 58939091 Ki = 14 nM T36483 C82PJI 59016133 Ki = 8 nM T36483 C4D0OU 59016136 Ki = 20 nM T36483 CNK7S5 59016155 Ki = 19.5 nM T36483 CX7GJ3 59110442 IC50 = 28 nM T36483 CQ70WI 59110450 IC50 = 22 nM T36483 CTE5W4 59110452 IC50 = 13 nM T36483 CNFW51 59110475 IC50 = 25 nM T36483 C1WUI8 59110479 IC50 = 33 nM T36483 CW5IM9 59110483 IC50 = 27 nM T36483 C2UTJ9 60003490 IC50 = 24 nM T36483 C8R2GE 70681077 IC50 = 8.8 nM T36483 CNV1K4 70683199 IC50 = 20 nM T36483 CH1QU9 70683205 IC50 = 8.6 nM T36483 CH1YU2 70683207 IC50 = 64 nM T36483 CRNG89 70685279 IC50 = 20 nM T36483 CP0K5B 70685280 IC50 = 35 nM T36483 CDHT12 70685282 IC50 = 49 nM T36483 CP67OG 70687423 IC50 = 225 nM T36483 CS7AR2 70687424 IC50 = 21 nM T36483 CE30ZT 70687425 IC50 = 513 nM T36483 CL78ZH 70687427 IC50 = 18 nM T36483 CIH25U 70693686 IC50 = 45 nM T36483 CN16RX 70695800 IC50 = 451 nM T36483 CTX46Q 71770951 IC50 > 30000 nM T36483 CK6EG1 72547305 IC50 = 1100 nM T36483 C1DEP5 72547306 IC50 = 220 nM T36483 CP6WG0 72547307 IC50 = 1.3 nM T36483 CU7L1V 72547308 IC50 = 210 nM T36483 CER7U3 72547551 IC50 = 7.2 nM T36483 CJLV20 72547552 IC50 = 26 nM T36483 CM5K7P 72547553 IC50 = 6 nM T36483 C5K1HR 72547554 IC50 = 50 nM T36483 CR89KZ 72547555 IC50 = 43 nM T36483 CEX78Z 72547556 IC50 = 2.7 nM T36483 CK87FB 73347045 EC50 = 110000 nM T36483 CJ9AL1 76285459 Ki = 5 nM T36483 C34FDW 76309941 IC50 = 2100 nM T36483 CY1TQ8 76309942 IC50 = 2000 nM T36483 C2XWP7 76310287 Ki = 239 nM T36483 C5MU6P 76310288 Ki = 12 nM T36483 CH4PG5 76310289 Ki = 24 nM T36483 C1R3JF 76310290 Ki = 25 nM T36483 CVL9M1 76313663 IC50 = 120 nM T36483 CQ4HY7 76313664 IC50 = 67 nM T36483 COMF86 76317165 IC50 = 280 nM T36483 CJO03F 76317166 IC50 = 360 nM T36483 C4OQ6V 76317512 Ki = 31 nM T36483 C3JBO9 76317513 Ki = 384 nM T36483 CQ54MK 76317514 Ki = 12.5 nM T36483 CU76WL 76324547 IC50 = 230 nM T36483 CH0DZ8 76324857 Ki = 13.5 nM T36483 CY4GX2 76328106 IC50 = 53 nM T36483 CV3BH9 76328107 IC50 = 33 nM T36483 COU9Q7 76328415 Ki = 14.5 nM T36483 C3SHJ4 76331783 IC50 = 7800 nM T36483 CCY2S9 76331784 IC50 = 230 nM T36483 C5HI1X 76332095 Ki = 98 nM T36483 CRW4D8 76332096 Ki = 32 nM T36483 C3U5BQ 76332097 Ki = 15 nM T36483 C3AFJ4 76335370 IC50 = 470 nM T36483 CN5AD3 76335371 IC50 = 980 nM T36483 CS43RT 76335372 IC50 = 67 nM T36483 CH01JU 76335711 Ki = 140 nM T36483 CU24GV 76335712 Ki = 180 nM T36483 C6Q7CA 76335713 Ki = 12.9 nM T36483 CIV74S 86302495 Ki = 5.1 nM T36483 CJ64EC 86302515 Ki = 8.9 nM T36483 C96WJL 90644636 Ki = 21 nM T36483 CIZK39 90644637 Ki = 15.5 nM T36483 C2Y9BG 90644638 Ki = 267 nM T36483 CK65RM 90644639 Ki = 26.5 nM T36483 COJ1Z8 90644640 Ki = 28 nM T36483 CB2F7G 90644641 Ki = 43 nM T36483 CRS60E 90644642 Ki = 25 nM T36483 CEWU84 90644643 Ki = 232 nM T36483 CN5YF3 90644644 Ki = 31.5 nM T36483 CML79P 90644645 Ki = 392 nM T36483 C1LHG8 90663288 IC50 = 23 nM T36483 CIZL42 90663289 IC50 = 270 nM T36483 C7RCD2 90663290 IC50 = 20 nM T36483 CR0G1L 90663291 IC50 = 46 nM T36483 CHZ9C1 90663292 IC50 = 40 nM T36483 CD9O6M 90663293 IC50 = 21.9 nM T36483 CP3BC7 90663294 IC50 = 250 nM T36483 CR7TN4 90663295 IC50 = 17 nM T36483 C0B1OR 90663296 IC50 = 870 nM T36483 CR40WY 90663297 IC50 = 32000 nM T36483 CUT54F 90663298 IC50 = 41 nM T36483 C2RVY5 90663299 IC50 = 500 nM T36483 C3S7PT 90663300 IC50 = 370 nM T36483 C37WFI 90663301 IC50 = 470 nM T36483 C3Z2BI 90663302 IC50 = 85000 nM T36483 CE5K8S 90663303 IC50 = 1000 nM T36483 CMB35Q 90663304 IC50 = 110 nM T36483 C2AIV3 90663305 IC50 = 64000 nM T36483 C8MBP2 90663306 IC50 = 34 nM T36483 CNP70T 90663307 IC50 = 99 nM T36483 CJB2G3 90663308 IC50 = 7600 nM T36483 CW5G6D 90663309 IC50 = 1180 nM T36483 CZW03D 90663310 IC50 = 320 nM T36483 CP37FV 90663311 IC50 = 28 nM T36483 CBRO21 90663312 IC50 = 200 nM T36483 C4UHS1 90663313 IC50 = 4 nM T36483 CUF1J9 90663314 IC50 = 16.6 nM T36483 C4V7TC 90663315 IC50 = 6.6 nM T36483 C43MOB 90663316 IC50 = 25 nM T36483 CSHL28 90663317 IC50 = 340 nM T36483 CV65ED 90663318 IC50 = 9 nM T36483 CEG37C 90663319 IC50 = 19 nM T36483 CR7Y3D 90663320 IC50 = 28 nM T36483 C0PHI2 90663321 IC50 = 130 nM T36483 CH7N5Y 90663322 IC50 = 500 nM T36483 C6X8QP 90663323 IC50 > 100000 nM T36483 C6T1GU 90663324 IC50 = 3440 nM T36483 CT15QB 90663325 IC50 = 42 nM T36483 CE2N9R 90663326 IC50 = 93 nM T36483 C8H3EK 90663327 IC50 = 39 nM T36483 CE7L2P 90663328 IC50 = 7.5 nM T36483 CI13QM 90663329 IC50 = 950 nM T36483 C1O8PU 90663330 IC50 = 40000 nM T36483 CMEZ14 90663331 IC50 = 680 nM T36483 CI8EF5 90663332 IC50 = 4670 nM T36483 C4W1ZL 90663333 IC50 = 3930 nM T36483 C4CN1K 90663334 IC50 = 110 nM T36483 C4S7IR 90663335 IC50 = 61 nM T36483 C2TI1O 90663336 IC50 = 630 nM T36483 CYXO35 90663337 IC50 = 21700 nM T36483 CEH10F 90663338 IC50 = 880 nM T36483 CMXW50 90663339 IC50 = 2320 nM T36483 CQO2T5 90663340 IC50 = 310 nM T36483 CL0MR2 90663341 IC50 = 350 nM T36483 CC9E6Y 90663342 IC50 = 9900 nM T36483 CE28ZM 90663343 IC50 = 1630 nM T36483 C0K6HW 90663344 IC50 = 260 nM T36483 CM6CH8 90663345 IC50 = 170 nM T36483 C8AD0J 90663346 IC50 = 24 nM T36483 CB1R3C 90663347 EC50 = 67000 nM T36483 CVZ0Q7 90663348 IC50 = 246 nM T36483 C9U6PF 90663350 IC50 = 340 nM T36483 CP8AT5 90663351 IC50 = 7550 nM T36483 CTV12X 90663352 IC50 = 1120 nM T36483 C2Y3KZ 90663353 IC50 = 4710 nM T36483 C5QR4T 90663354 IC50 = 560 nM T36483 C7XQS8 90663355 IC50 = 24 nM T36483 C1IEB4 90663356 IC50 = 2730 nM T36483 CH0I1E 90663358 IC50 = 66700 nM T36483 C8T4KN 90663359 EC50 = 270 nM T36483 CJ2PY5 90663360 IC50 = 220 nM T36483 COS70P 90663563 IC50 = 1190 nM T36483 C50FEG 90663732 IC50 = 19 nM T36483 CE5V6U 117072551 IC50 = 1700 nM T36483 CNS91H 117909194 IC50 = 28.7 nM T36483 CR07ZG 117909666 IC50 = 4.22 nM T36483 C6N8SM 117909768 IC50 = 3.08 nM T36483 C4OVE8 118714099 IC50 > 10000 nM T36483 CC4LA1 118953461 IC50 > 30000 nM T36483 C13EIL 118967091 IC50 > 30000 nM T36483 C5OKW0 118967130 IC50 > 30000 nM T36483 CE3CN6 118971057 IC50 > 30000 nM T36483 CT4RP7 118971061 IC50 > 30000 nM T36483 CD7AN0 118971371 IC50 > 30000 nM T36483 CQD4P5 121469330 IC50 = 0.99 nM T36483 C5Y7VT 125407509 IC50 > 30000 nM T36483 CW03MF 126961335 IC50 > 50000 nM T36483 CDR2I3 127049415 IC50 = 100 nM T36483 C2UJ0N 127050656 IC50 = 60 nM T36483 C2V5EI 127050657 IC50 = 10 nM T36483 CYBO14 127050658 IC50 = 50 nM T36483 CK7U9R 127050672 IC50 = 130 nM T36483 CF6M7Y 127050673 IC50 = 30 nM T36483 CE80LC 127050934 IC50 = 30 nM T36483 C2ENH5 127050971 IC50 = 40 nM T36483 C31MDQ 127051545 IC50 = 60 nM T36483 C9YT7Q 127051546 IC50 = 70 nM T36483 CD2LB1 127051547 IC50 = 80 nM T36483 CUO21P 134137936 IC50 > 10000 nM T36483 CP12TG 136209460 IC50 ~ 90000 nM T36483 CU67ND 137631870 IC50 = 9500 nM T36483 CK38CP 137632009 IC50 = 3000 nM T36483 C7XYM6 137632193 IC50 = 12000 nM T36483 C6KND9 137632824 IC50 > 100000 nM T36483 C21SWT 137632975 IC50 = 8700 nM T36483 C61BPT 137633371 IC50 = 32000 nM T36483 CE3WA8 137634922 IC50 > 100000 nM T36483 CPY6H8 137635753 IC50 > 100000 nM T36483 C3TI7G 137637794 IC50 = 14000 nM T36483 CGF2X7 137638549 IC50 = 19000 nM T36483 CZ0T3W 137638930 IC50 > 100000 nM T36483 C50LQS 137639606 IC50 = 20000 nM T36483 C5R9AQ 137641036 IC50 > 100000 nM T36483 CA60IO 137641321 IC50 > 100000 nM T36483 CCUE34 137642658 IC50 > 100000 nM T36483 C4WEG7 137643571 IC50 > 100000 nM T36483 C1F4YR 137644873 IC50 = 55000 nM T36483 CSP79Y 137645208 IC50 = 1500 nM T36483 C2VK3O 137645447 IC50 > 100000 nM T36483 CH6JZ5 137647264 IC50 = 23000 nM T36483 CTS03I 137648050 IC50 > 100000 nM T36483 CO6ZT4 137649563 IC50 = 7000 nM T36483 C14CLO 137649807 IC50 > 100000 nM T36483 CY7VL5 137651100 IC50 > 100000 nM T36483 CYU8K1 137651696 IC50 > 100000 nM T36483 C8V7XZ 137652024 IC50 = 87000 nM T36483 CDA2K4 137652763 IC50 > 100000 nM T36483 CCZY19 137653180 IC50 = 8100 nM T36483 C5YMI9 137653221 IC50 > 100000 nM T36483 CR6TX5 137653750 IC50 = 14000 nM T36483 C8B4DQ 137654003 IC50 > 100000 nM T36483 C91MIW 137654212 IC50 = 21000 nM T36483 C2E9JM 137654568 IC50 = 29000 nM T36483 CF4S7T 137654736 IC50 > 100000 nM T36483 CM2HE5 137655130 IC50 = 10000 nM T36483 CG07RC 137656188 IC50 > 100000 nM T36483 C8AZ7S 137657212 IC50 > 100000 nM T36483 CZP1K2 137657357 IC50 > 100000 nM T36483 CCX5T7 137658131 IC50 > 100000 nM T36483 C10QES 137658217 IC50 > 100000 nM T36483 CP1QS4 137659611 IC50 = 9100 nM T36483 CIW4T5 137660576 IC50 > 100000 nM T36483 C0YHD2 137661486 IC50 = 650 nM T36483 CCU4J5 137661676 IC50 = 17000 nM T36483 CB3HI7 145967675 IC50 > 10000 nM T36483 CF4V1J 145968568 IC50 = 19.95 nM T36483 CW70RF 145970191 IC50 = 290 nM T36483 CTEJ01 145971090 IC50 = 100000 nM T36483 CKVH05 154688304 IC50 = 398.11 nM T36483 COY7A6 154688307 IC50 = 370 nM T36483 CPX6Q0 155512671 IC50 = 40 nM T36483 CNY3Z8 155519325 IC50 = 398.11 nM T36483 C5CJF2 155526775 IC50 = 10 nM T36483 CQN9L7 155536026 IC50 = 30 nM T36483 CFDM94 155549751 IC50 = 140 nM T36483 CN4WT6 155564785 IC50 = 130 nM T36483 CHY4T0 44306337 IC50 = 150 nM T36483 C2DVJ6 44306349 IC50 = 6100 nM T36483 D00KRL 10132921 IC50 > 10000 nM T36483 D0BV3B 16214871 Ki = 19 nM T36483 D0I2VE 9853822 IC50 = 440 nM T36483 D0QK2E 9804049 Ki = 2.7 nM T12797 D02OZK 11404337 EC50 = 600 nM T12797 D03TTE 135513044 Ki = 1470 nM T12797 D0B1UL 136002683 Ki = 460 nM T12797 D0CR9A 136183441 Ki = 930 nM T12797 D0L8WH 11228183 Ki > 20000 nM T12797 CVD64E 36941 Ki > 100000 nM T12797 CB6E4Y 720528 IC50 = 2100 nM T12797 C2I9CA 779754 IC50 = 300 nM T12797 CBO6D7 1074953 IC50 = 450 nM T12797 C87OXF 1180669 IC50 > 50000 nM T12797 C4Y5CT 1180675 IC50 > 50000 nM T12797 COW3Q9 1180676 IC50 = 600 nM T12797 CGAM30 1582605 Ki = 6140 nM T12797 C07WVL 1654287 IC50 = 4100 nM T12797 CW2UC7 1664226 IC50 = 2400 nM T12797 CJ5FD3 1673604 IC50 = 2600 nM T12797 CN96HL 2268888 IC50 > 10000 nM T12797 C4LM7K 16654625 IC50 > 50000 nM T12797 CMO71D 16654638 IC50 = 8700 nM T12797 C3S2BO 16654639 IC50 = 11100 nM T12797 C8AYR4 16654640 IC50 = 1000 nM T12797 CG8IE3 16654650 IC50 > 10000 nM T12797 CVWX79 16654652 IC50 = 400 nM T12797 C8INE7 16654653 IC50 = 600 nM T12797 CLT31W 16654654 IC50 = 1100 nM T12797 C3K7AN 16654655 IC50 = 690 nM T12797 CR93CM 16654656 IC50 = 1700 nM T12797 CY3D6Z 16654661 IC50 = 2100 nM T12797 CL3BH9 16654662 IC50 = 1300 nM T12797 C6NH0G 16654665 IC50 > 10000 nM T12797 CTZS48 16654669 IC50 = 620 nM T12797 CKX1T5 16654670 IC50 = 6200 nM T12797 CH4C1D 16654672 IC50 = 8300 nM T12797 CC76JQ 16654674 IC50 = 10500 nM T12797 C8EIO1 16654677 IC50 = 1200 nM T12797 CD6YT8 16654679 IC50 = 2000 nM T12797 CX1JA7 16654730 IC50 = 10800 nM T12797 CY5UW9 16654772 IC50 = 3900 nM T12797 CXO2S9 44191694 IC50 = 550 nM T12797 CHT92S 44191696 IC50 = 1300 nM T12797 C83UCJ 44191750 IC50 = 670 nM T12797 CMS39X 44191815 IC50 = 5000 nM T12797 C0J3RT 44192144 IC50 = 400 nM T12797 C97RQU 44192145 IC50 = 2000 nM T12797 C57VCY 44224066 IC50 = 730 nM T12797 CH2E4R 44609307 Ki = 2340 nM T12797 CG2NH7 46236925 IC50 = 590 nM T12797 C78NZA 46236926 IC50 = 770 nM T12797 CUB3N9 52943093 IC50 = 29000 nM T12797 C8C7FS 71451698 EC50 = 25500 nM T12797 CJA8N4 71455243 EC50 = 8200 nM T12797 COH24E 71455246 EC50 = 17800 nM T12797 CVC5F8 71455247 EC50 = 21500 nM T12797 CUG8N7 71462421 EC50 = 24000 nM T12797 CP3Y2O 71548702 Ki = 1110 nM T12797 CS02CG 71549001 Ki = 3180 nM T12797 C37AJW 71549412 Ki = 17260 nM T12797 C3C7QO 86765310 Ki = 3360 nM T12797 C5W2EA 118734957 Ki > 660 nM T12797 C76SBJ 122622651 Ki = 3700 nM T12797 CR19KU 122622656 Ki = 900 nM T12797 CFR02M 122622711 Ki = 170 nM T12797 CY2J6L 122622713 Ki = 1700 nM T12797 C0AYP2 122622799 Ki = 3000 nM T12797 CE4MG7 122622800 Ki = 1600 nM T12797 C0KP5W 122622803 Ki = 810 nM T12797 CIH4M1 122622824 Ki = 3800 nM T12797 CBFO10 122622827 Ki = 760 nM T12797 C6JOM4 122622922 Ki = 3400 nM T12797 CY9OL2 122623097 Ki = 570 nM T12797 C59MST 122623143 Ki = 150 nM T12797 C9YU0H 122623413 Ki = 1000 nM T12797 CJ5P7N 122623425 Ki = 4600 nM T12797 C1R4UJ 122633925 Ki = 1100 nM T12797 C26QUL 122633937 Ki = 14800 nM T12797 CB4J7Z 134130355 Ki < 0.1 nM T12797 CC9OV6 134131166 Ki = 32 nM T12797 C9MFV2 136002682 Ki = 870 nM T12797 C6FY0E 136002684 Ki = 470 nM T12797 C9RD0X 136032611 Ki = 470 nM T12797 CC09EN 136183442 Ki = 9330 nM T12797 CYJD84 136183443 Ki = 3530 nM T12797 CF8HV7 136183446 IC50 = 122 nM T12797 CCVP03 145994390 Ki = 100 nM T12797 C1R8MS 155522698 Ki = 390 nM T12797 C5L4DX 155523696 Ki = 250 nM T12797 CQN1B8 155524663 Ki > 70000 nM T12797 CB89NA 155528220 Ki > 70000 nM T12797 CU9CX1 155529604 Ki = 280 nM T12797 CUS28M 155542793 Ki = 84 nM T12797 CVBF96 155545115 Ki = 10600 nM T12797 CL4HF7 155547093 Ki = 100 nM T12797 C4KGR1 155556368 Ki = 62000 nM T12797 D05RDP 992586 Ki = 5330 nM T12797 D0V7PX 454878 IC50 > 10000 nM T60897 D05EAM 4735 IC50 = 300 nM T60897 CPQ3D4 1202786 IC50 = 188000 nM T60897 C9C0OM 2714312 IC50 = 31400 nM T60897 C85XHT 7509342 IC50 = 69400 nM T60897 CYOS08 8119828 IC50 = 104000 nM T60897 C3NIY8 16456878 IC50 = 188000 nM T60897 CBXR07 45840460 IC50 = 149800 nM T60897 CEL91T 56923561 IC50 = 109200 nM T60897 C2IT1Z 91383855 IC50 = 277 nM T60897 CU3RP8 124141953 IC50 = 52 nM T71266 D01NEC 51042438 IC50 = 1.3 nM T71266 D01ZAQ 25227436 IC50 = 8 nM T71266 D02NNV 3038525 IC50 > 5000 nM T71266 D02ZQS 16095342 IC50 = 1510 nM T71266 D09IYM 24905401 IC50 = 50 nM T71266 D0E3TC 44259 IC50 = 5 nM T71266 D0I4TH 24788740 IC50 = 8 nM T71266 D0MS3Z 16725726 IC50 = 9 nM T71266 D0W3RW 24964624 IC50 = 65 nM T71266 D03BNU 59604787 IC50 > 10000 nM T71266 D0T3ME 156422 IC50 > 30000 nM T71266 CWN6P7 5702541 IC50 = 662 nM T71266 CG17TN 6914611 IC50 = 35 nM T71266 C7E2QK 6914613 IC50 = 354 nM T71266 CIAL53 9819282 IC50 > 50000 nM T71266 C41QWA 9857146 IC50 > 10000 nM T71266 CI0AW6 9871034 IC50 = 27000 nM T71266 CS5KX9 9938299 IC50 > 10000 nM T71266 CJX43Z 10055074 IC50 = 7400 nM T71266 C7TA9J 10113568 IC50 = 17378.01 nM T71266 CEV18B 10128689 IC50 > 50000 nM T71266 C7PK4U 10152003 IC50 > 50000 nM T71266 C4FUG5 10152760 IC50 > 50000 nM T71266 CMO32F 10152761 IC50 = 21870 nM T71266 CMR17F 10174144 IC50 > 50000 nM T71266 CLP79V 10196532 IC50 = 3200 nM T71266 CI8MW4 10216627 IC50 = 73 nM T71266 C0O8FI 10217663 IC50 = 33100 nM T71266 CY6MJ3 10218178 IC50 > 50000 nM T71266 C8V6RI 10240275 IC50 = 7200 nM T71266 CD3W6Y 10289038 IC50 > 50000 nM T71266 C2LP9A 10289671 IC50 = 2400 nM T71266 C4MOF8 10312133 IC50 = 1613 nM T71266 CAK9U4 10415819 IC50 = 1228 nM T71266 C2ON6C 11246455 IC50 = 179 nM T71266 C49NET 11256399 IC50 = 380 nM T71266 C6C3JX 11281930 IC50 > 10000 nM T71266 CBOP58 11293798 Ki = 4890 nM T71266 C5ACQ0 11348837 IC50 = 3000 nM T71266 C26BZX 11362471 Ki > 10000 nM T71266 CWXB93 11397177 Ki > 10000 nM T71266 CVG3L6 11502369 IC50 = 990 nM T71266 CK2WT3 11510023 IC50 = 1500 nM T71266 CL2I5O 11517293 IC50 = 19000 nM T71266 C05MTD 11522988 IC50 = 4700 nM T71266 C8IHX9 11538014 IC50 = 5400 nM T71266 CTG83F 11539329 Ki > 9500 nM T71266 CBIY48 11544625 IC50 = 5000 nM T71266 C2QDA9 11559783 IC50 = 2900 nM T71266 CACS26 11561968 Ki > 2000 nM T71266 C9THO1 11567357 IC50 = 610 nM T71266 CW4Z9E 11575743 IC50 = 280 nM T71266 CMIL86 11590363 Ki > 9500 nM T71266 C4Z1YB 11610430 IC50 = 1100 nM T71266 C9T6SC 11640926 Ki > 9500 nM T71266 C7XEV0 11664023 IC50 = 2474 nM T71266 CJB19K 11667833 IC50 = 18000 nM T71266 C0V7SU 11675388 IC50 = 57 nM T71266 CU0E8O 11690457 Ki > 10000 nM T71266 CDF53M 11718648 IC50 = 2600 nM T71266 C9A6KM 11857236 IC50 = 3 nM T71266 C39VTW 11959283 IC50 = 70 nM T71266 C36HDX 11959286 IC50 = 30 nM T71266 CO0A4K 11959314 IC50 = 1 nM T71266 C12CRJ 11959377 IC50 = 22 nM T71266 C1WDQ0 11959682 IC50 = 49 nM T71266 CMW89V 11959683 IC50 = 17 nM T71266 C7N6CQ 15604547 IC50 = 76 nM T71266 CFPW41 16007116 Ki > 9500 nM T71266 CZK8V6 16043304 IC50 = 2.6 nM T71266 C9TU1O 16046126 IC50 > 1000 nM T71266 C7Z4LV 16095343 IC50 = 1290 nM T71266 C54YXC 16121514 IC50 = 72.44 nM T71266 CJXU82 21103111 IC50 > 50000 nM T71266 CF9YE6 21103119 IC50 > 50000 nM T71266 C5AR9M 21103197 IC50 > 50000 nM T71266 CN1O7X 23647016 IC50 > 50000 nM T71266 CJ3EO0 23647017 IC50 = 3973 nM T71266 CH14KD 23647018 IC50 > 50000 nM T71266 CQ5Z0J 23647019 IC50 > 50000 nM T71266 C2JTA3 23647573 IC50 = 39 nM T71266 C7YG1N 24759534 IC50 > 100000 nM T71266 CW3JR8 24783593 IC50 = 10 nM T71266 C05MQY 24783594 IC50 = 23 nM T71266 C93TIM 24786152 IC50 = 5 nM T71266 CSY9Z6 24788164 IC50 = 10 nM T71266 CFR62V 24788432 IC50 = 5 nM T71266 C2JNI3 24788623 IC50 = 13 nM T71266 CMR7F1 24788739 IC50 = 5 nM T71266 CY1ZS7 24803305 IC50 = 2 nM T71266 C2ANO6 24804134 IC50 = 3 nM T71266 CSH8A5 24804780 IC50 = 3 nM T71266 CUTH13 24805273 IC50 = 20 nM T71266 CA9F3Y 25023714 IC50 = 398 nM T71266 C8Z4PI 25023715 IC50 = 1410 nM T71266 CV96QX 25023716 IC50 = 1290 nM T71266 C5INV4 25023717 IC50 = 1549 nM T71266 CPOH02 25023718 IC50 = 3020 nM T71266 C6F7RD 25023719 IC50 = 2290 nM T71266 C1JEU6 25023729 IC50 = 69 nM T71266 CR8JP7 25023735 IC50 = 9 nM T71266 C4W7LY 25023736 IC50 = 16 nM T71266 COV3Q4 25061501 IC50 = 12 nM T71266 C8NR9H 25170562 IC50 = 5 nM T71266 CS9LC3 25170563 IC50 = 12 nM T71266 CN8YZ4 25170991 IC50 = 26 nM T71266 CSY93F 25190765 IC50 > 1000000 nM T71266 C0BCX6 25190766 IC50 = 1610 nM T71266 C19TVC 25190767 IC50 = 774 nM T71266 CK9V3Y 25190768 IC50 = 56.6 nM T71266 CD7S6Q 25190770 IC50 = 3750 nM T71266 C3HU6A 25190771 IC50 = 2.38 nM T71266 CHN5O0 25190977 IC50 = 2 nM T71266 COWB90 25221040 IC50 = 6 nM T71266 CC25TV 25222706 IC50 = 3 nM T71266 C1IG7E 25243798 IC50 > 10000 nM T71266 CH65JV 25243799 IC50 > 10000 nM T71266 CBQO98 42602095 IC50 = 30 nM T71266 CJ61SE 42602096 IC50 = 15 nM T71266 CI42XG 42602097 IC50 = 24 nM T71266 CD2AH4 42602175 IC50 = 22 nM T71266 CSWA85 42602176 IC50 = 40 nM T71266 C1LUN4 42602178 IC50 = 7 nM T71266 C8O3EA 42602260 IC50 = 15 nM T71266 C93NKL 42602264 IC50 = 4 nM T71266 C5OHU9 44414317 IC50 = 5200 nM T71266 CBO18Y 44414320 IC50 = 660 nM T71266 CWD30R 44414422 IC50 = 240 nM T71266 C25ZRP 44414445 IC50 > 25000 nM T71266 CW4HT5 44414446 IC50 > 25000 nM T71266 CCH43E 44414447 IC50 = 11 nM T71266 C4FI1S 44414467 IC50 > 25000 nM T71266 C2CE5X 44414470 IC50 = 27 nM T71266 CI2G5K 44414471 IC50 = 1300 nM T71266 C93QFH 44414472 IC50 = 7000 nM T71266 CTDY95 44414507 IC50 = 1000 nM T71266 CY58PE 44414508 IC50 > 25000 nM T71266 C91ZIP 44414529 IC50 = 2800 nM T71266 CI26HQ 44414530 IC50 = 820 nM T71266 CIMY48 44414553 IC50 = 2400 nM T71266 C3JHE6 44414577 IC50 > 25000 nM T71266 C0E4CL 44414579 IC50 = 4.8 nM T71266 C1FU3D 44414608 IC50 > 25000 nM T71266 C6R9AN 44414634 IC50 = 2300 nM T71266 CQB9Z0 44414635 IC50 > 25000 nM T71266 CYX64I 44414652 IC50 = 2100 nM T71266 CC21KN 44414653 IC50 = 7400 nM T71266 CQ93OC 44414655 IC50 > 25000 nM T71266 COP8A3 44449880 IC50 = 1900 nM T71266 CDEJ84 44450004 IC50 = 11280 nM T71266 C8OG1V 44517709 IC50 = 4000 nM T71266 C0DJS1 44591843 IC50 = 2 nM T71266 CX52YW 44591844 IC50 = 1 nM T71266 C1LS6V 44591845 IC50 = 3 nM T71266 CSZ5R9 44592438 IC50 = 40 nM T71266 CTS95L 44592502 IC50 = 2 nM T71266 CSKZ16 44592503 IC50 = 2 nM T71266 COY57J 44592504 IC50 = 2 nM T71266 C3CDV8 44592505 IC50 = 2 nM T71266 CAZE46 46175126 IC50 = 270 nM T71266 CQ5SD4 46190876 IC50 = 10 nM T71266 CY3HW5 46224684 IC50 = 1100 nM T71266 CB5H9C 46225574 IC50 = 15 nM T71266 C8M1DT 46225589 IC50 = 1 nM T71266 C60XUQ 46226079 IC50 = 1 nM T71266 C5PCH8 46226080 IC50 = 2 nM T71266 C6UD1Y 46226095 IC50 = 19 nM T71266 C7IF4T 46226096 IC50 = 10 nM T71266 CUDZ46 46226135 IC50 = 500 nM T71266 C0P4CT 46226136 IC50 = 2 nM T71266 CPH49S 46226137 IC50 = 1 nM T71266 CM5X8B 46226156 IC50 = 1 nM T71266 CLS29B 46872626 IC50 > 10000 nM T71266 C3HG7B 46882134 IC50 = 900 nM T71266 CTSE94 46882135 IC50 = 4600 nM T71266 CSY9H1 46882136 IC50 = 27000 nM T71266 CO16JL 46882137 IC50 = 12 nM T71266 CJEM76 46882138 IC50 = 42 nM T71266 CRZ91X 46882835 IC50 = 360000 nM T71266 CS0V9G 46882836 IC50 = 28000 nM T71266 CU8WX3 46882837 IC50 = 900000 nM T71266 C2O8RZ 46886323 IC50 > 1000 nM T71266 C70BLN 46886550 IC50 = 65 nM T71266 CCV96R 46886665 IC50 = 43 nM T71266 CC1Y0M 52941299 IC50 = 5769 nM T71266 CDT94U 52941495 IC50 = 2056 nM T71266 C9UF6K 52941555 IC50 = 485 nM T71266 CYM80Q 52942489 IC50 = 13916 nM T71266 CS09YT 52942516 IC50 = 6073 nM T71266 CQ08WT 52942668 IC50 = 1122 nM T71266 CHW04J 52943916 IC50 = 754 nM T71266 CY8BV4 52944892 IC50 = 746 nM T71266 CEM95A 52946401 IC50 = 6079 nM T71266 CKE3C7 52946402 IC50 = 1464 nM T71266 C3Q4CU 52947490 IC50 = 8410 nM T71266 CR9E1Z 52947590 IC50 = 25110 nM T71266 CE81HA 52950003 IC50 = 363 nM T71266 C3TU8R 52950063 IC50 = 666 nM T71266 C7MC5G 52950205 IC50 = 2718 nM T71266 C8NA4L 53384644 IC50 > 30000 nM T71266 CPC5D2 56603995 IC50 = 40 nM T71266 CS7U9L 56965952 IC50 = 170 nM T71266 CQP7E0 57750290 IC50 = 18 nM T71266 CNBO65 57750312 IC50 = 30 nM T71266 C2F9DS 57750315 IC50 = 105 nM T71266 CZ08KN 57750321 IC50 = 36 nM T71266 CUY8T6 57750329 IC50 = 582 nM T71266 CK4W1L 57750342 IC50 = 10 nM T71266 CM5X9L 57750343 IC50 = 523 nM T71266 CBY5E4 57750369 IC50 = 15 nM T71266 CSI9Y4 57750382 IC50 = 270 nM T71266 C6GH7X 57750391 IC50 = 150 nM T71266 CL7CW0 57750402 IC50 = 100 nM T71266 CA4G5W 57750407 IC50 = 6 nM T71266 CM7XL6 57750408 IC50 = 16 nM T71266 CY4Z8R 57750418 IC50 = 176 nM T71266 C87LKR 58191080 IC50 = 3 nM T71266 CZPF92 58191081 IC50 = 2 nM T71266 CZA32V 58344912 IC50 = 22000 nM T71266 CPVF85 58344916 IC50 = 24000 nM T71266 CD3LX9 58344922 IC50 = 700 nM T71266 CS8ZY7 58344924 IC50 = 390 nM T71266 C89NVR 58344941 IC50 = 170 nM T71266 CYK74H 58344983 IC50 = 370 nM T71266 CRJ47B 58345005 IC50 = 71000 nM T71266 CIOV02 58345019 IC50 > 100000 nM T71266 CY62SG 58345029 IC50 = 660 nM T71266 CM5HE1 58345070 IC50 > 10000 nM T71266 CO18NP 58345151 IC50 = 390 nM T71266 CV61YJ 58345169 IC50 > 100000 nM T71266 CW6SC9 58345215 IC50 > 100000 nM T71266 CFLZ87 58345232 IC50 = 2500 nM T71266 CYBT41 58345302 IC50 = 660 nM T71266 C4PE7X 58345314 IC50 = 400 nM T71266 C8X3WB 58458198 IC50 = 4160 nM T71266 C20XPF 58458267 IC50 > 2000 nM T71266 CP85TJ 58458278 IC50 = 1 nM T71266 CT79LH 58458379 IC50 = 83 nM T71266 CXJ63M 59603829 IC50 > 100000 nM T71266 CQEU96 59603842 IC50 = 330 nM T71266 CPVD45 59670809 IC50 = 21 nM T71266 C32WHR 59670989 IC50 = 12 nM T71266 CDWQ04 59671004 IC50 = 28 nM T71266 C43HZT 59671085 IC50 = 73 nM T71266 C0BRA5 59671144 IC50 = 45 nM T71266 CEYW16 59671148 IC50 = 4 nM T71266 C50NWX 59671151 IC50 = 2 nM T71266 CZH4W5 59671179 IC50 = 7 nM T71266 C8FY0G 59671180 IC50 = 7 nM T71266 C1MR8Q 60097495 IC50 > 2500 nM T71266 CC3MB4 60155179 IC50 > 100000 nM T71266 C9QB8G 60155270 IC50 = 2600 nM T71266 CM6NF2 60155627 IC50 > 10000 nM T71266 C62SQG 60155628 IC50 = 86 nM T71266 COS39T 60155629 IC50 = 430 nM T71266 CV63UL 67240318 IC50 > 10000 nM T71266 CP8OI2 67304551 IC50 > 10000 nM T71266 CY76UR 67305743 IC50 = 8.1 nM T71266 C3UKG8 67312397 IC50 = 5.4 nM T71266 CM6TZ3 67312506 IC50 = 26 nM T71266 C5DGR9 69036886 IC50 = 10000 nM T71266 CS8UF1 70675988 IC50 = 5 nM T71266 C2W5BX 70675991 IC50 = 798 nM T71266 CUJA60 70676312 IC50 = 4 nM T71266 CRBW21 70676316 IC50 = 27 nM T71266 CGX49K 70676464 IC50 = 3 nM T71266 C5D1LV 70687790 IC50 = 9120.11 nM T71266 CKT60L 71455860 Ki > 9000 nM T71266 CQV96E 71583048 IC50 = 4260 nM T71266 CSPR52 71583049 IC50 = 8065 nM T71266 CNT5F3 71583050 IC50 = 756 nM T71266 CH7I0W 71583051 IC50 = 2893 nM T71266 CJ2T9E 76332983 IC50 > 10000 nM T71266 C1HW4B 89735655 IC50 = 2400 nM T71266 C8GZ2B 135449326 Ki = 1800 nM T71266 CC73PA 138911338 IC50 = 1.7 nM T71266 CSU93V 155077019 IC50 = 0.12 nM T71266 C2MD1Q 155513187 IC50 > 10000 nM T71266 CL5DR0 155525783 IC50 = 0.1 nM T71266 CHS21A 155553831 IC50 = 65 nM T71266 CG95WV 155563831 IC50 = 4 nM T71266 CEIW13 155566807 IC50 = 700 nM T71266 D00ERW 44444843 Ki = 7157 nM T71266 D00HVA 11624601 Ki > 9500 nM T71266 D05APZ 135398501 IC50 > 2119 nM T71266 D05JRA 25190769 IC50 = 14.6 nM T71266 D09FFE 449241 IC50 = 200 nM T71266 D0I1FJ 11393719 IC50 = 646 nM T71266 D0J3LR 11634725 Ki > 4000 nM T71266 D0L2WP 46225540 IC50 = 1 nM T71266 D0OX1T 10172943 IC50 = 51 nM T71266 D0Q3NG 11715520 Ki > 9500 nM T71266 D0S7IE 11658882 Ki > 9500 nM T99948 D0OK1S 117941742 IC50 = 146 nM T99948 D0WQ9X 117951478 IC50 = 18 nM T99948 C1RCQ7 117941376 IC50 = 110 nM T99948 C7BVK6 117941458 IC50 = 1010 nM T99948 C6AL2M 117941533 IC50 = 6 nM T99948 C03JDG 117941658 IC50 = 6 nM T99948 CG3T5I 117941713 IC50 = 6 nM T99948 CL56TV 117941821 IC50 = 6 nM T99948 CYH13Z 117941887 IC50 = 80 nM T99948 CD0QR5 118434635 IC50 = 1.4 nM T99948 C4N1MD 121452782 IC50 = 6 nM T99948 C7P6CO 131839624 IC50 = 2.25 nM T99948 C2X0IF 145992098 IC50 = 5.2 nM T99948 D02BZV 91663303 IC50 = 6 nM T66538 D09BVL 4552 IC50 = 5888.44 nM T66538 D0S6QR 214350 EC50 = 352 nM T66538 CY1Z5T 232768 IC50 = 15135.61 nM T66538 CZU3E2 459332 IC50 = 13489.63 nM T66538 CEH76V 483833 IC50 = 18620.87 nM T66538 C7VH5Q 483836 IC50 = 17378.01 nM T66538 C7X9HU 740278 IC50 = 11748.98 nM T66538 CD5ZH7 830720 IC50 = 30199.52 nM T66538 C1UWX0 837857 IC50 = 26915.35 nM T66538 CFZ4U5 839448 IC50 = 11220.18 nM T66538 C3E4FV 868972 IC50 = 12302.69 nM T66538 C10NVJ 1124061 IC50 = 30902.95 nM T66538 CDOR89 1234642 IC50 = 12589.25 nM T66538 CU2FW1 2798242 IC50 = 3090.3 nM T66538 CLS15O 2798243 IC50 = 3467.37 nM T66538 CXW6L7 2946791 IC50 = 691.83 nM T66538 CTD1P7 2953683 IC50 = 3090.3 nM T66538 CU4P0Z 3011444 IC50 = 30902.95 nM T66538 CB0NG4 3011445 IC50 = 15135.61 nM T66538 C2MTJ0 3011446 IC50 = 11748.98 nM T66538 C0D3AK 3491594 IC50 = 19498.45 nM T66538 CL82TS 3605484 IC50 = 2511.89 nM T66538 C7Q9TV 4050379 IC50 = 251.19 nM T66538 CND86W 5073804 IC50 = 9332.54 nM T66538 CPW4Y1 9815734 EC50 = 8120 nM T66538 CJGX96 9881289 EC50 = 5070 nM T66538 CLHQ23 9990728 IC50 = 17782.79 nM T66538 C0T8UE 10035337 EC50 = 5130 nM T66538 CAQW79 10038562 EC50 = 4430 nM T66538 C6BEY4 10064074 IC50 = 3.236 nM T66538 C0GQF7 10083014 EC50 = 3340 nM T66538 C2CGW9 10243969 IC50 = 144.54 nM T66538 CQ8G6K 10263172 EC50 = 3860 nM T66538 C05UVN 10263770 EC50 = 15100 nM T66538 CJY45S 10331385 IC50 = 112201.85 nM T66538 CI1P3F 10354434 EC50 = 6750 nM T66538 C9N3KR 10356396 IC50 = 2630.27 nM T66538 CDFW74 10398337 EC50 = 6940 nM T66538 CX1SL4 10444440 IC50 = 13803.84 nM T66538 CUO6A4 10469103 EC50 = 17000 nM T66538 CS0OM5 10515414 IC50 = 154881.66 nM T66538 CF5I6P 10634209 IC50 = 93325.43 nM T66538 C9HG2C 10660593 IC50 = 24547.09 nM T66538 CG8W9V 10709096 IC50 = 37153.52 nM T66538 CI4P9O 10729882 IC50 = 93325.43 nM T66538 CN9KY8 10778936 IC50 = 28183.83 nM T66538 CU0BP4 10800545 IC50 = 104712.85 nM T66538 C5JQ8A 10849039 IC50 = 18620.87 nM T66538 CL8IW0 10849172 IC50 = 54954.09 nM T66538 C56UXE 10903109 IC50 = 79432.82 nM T66538 CX7S5A 10967695 IC50 = 2454.71 nM T66538 C0DS8B 10968747 IC50 = 8709.64 nM T66538 C5YA6S 10969679 IC50 = 5888.44 nM T66538 C8GK5I 11000844 IC50 = 6918.31 nM T66538 C2G6LX 11042812 IC50 = 1548.82 nM T66538 C7TDS2 11065065 IC50 = 3019.95 nM T66538 C6U8KG 11108600 IC50 = 10964.78 nM T66538 COF9D1 11109578 IC50 = 2137.96 nM T66538 CA38LS 11254734 IC50 = 190.55 nM T66538 CZ7K3W 11335564 IC50 = 7762.47 nM T66538 CL01DC 11392406 IC50 = 645.65 nM T66538 CCV2U0 11437030 IC50 = 27.54 nM T66538 C1GZ8U 11471747 IC50 = 446.68 nM T66538 C7O3AF 11472034 IC50 = 371.54 nM T66538 C3BI1D 11536112 IC50 = 10232.93 nM T66538 CRP35C 11651603 IC50 = 13489.63 nM T66538 C59YUQ 11779066 IC50 = 27.54 nM T66538 CJ58MG 11782023 IC50 = 3311.31 nM T66538 COM63L 11818496 IC50 = 177.83 nM T66538 CFJ3I2 11820396 EC50 = 5860 nM T66538 C1MZQ9 11823359 IC50 = 54954.09 nM T66538 CR72ZX 15717694 IC50 = 1445.44 nM T66538 CM7J9B 16099761 IC50 = 4073.8 nM T66538 CX2MQ8 16099762 IC50 = 5248.07 nM T66538 CKS0L7 16099763 IC50 = 30199.52 nM T66538 CTHR97 16099764 IC50 = 11748.98 nM T66538 CD3Q8R 16099767 IC50 = 11220.18 nM T66538 C7LAE8 18103922 IC50 = 15848.93 nM T66538 C7CZD5 24285062 IC50 = 134.9 nM T66538 C7EI0Y 24285063 IC50 = 8128.31 nM T66538 C8PTB6 44570449 IC50 = 281.84 nM T66538 CK2G5D 136029155 EC50 = 13400 nM T08123 D0R0MW 5329102 IC50 = 28 nM T08123 D08ZPO 448043 IC50 = 244 nM T08123 D0E3TC 44259 IC50 = 1 nM T08123 D0H2HZ 60194098 IC50 = 3981.07 nM T08123 D0HY9S 73386890 IC50 = 48 nM T08123 CY13DC 360689 IC50 = 5760 nM T08123 CCX69G 580694 IC50 = 100 nM T08123 CD5NJ1 953496 IC50 = 520 nM T08123 C6XYA1 953540 IC50 = 4460 nM T08123 CCN24W 1563747 IC50 = 2000 nM T08123 C3GZ8M 2358577 IC50 = 10000 nM T08123 CA6F4S 2360386 IC50 = 10000 nM T08123 CR09XN 2410620 IC50 = 194 nM T08123 C38OMQ 2727431 IC50 = 173 nM T08123 C85TOM 2727432 IC50 = 50 nM T08123 CI6H0F 2727439 IC50 = 1555 nM T08123 C3T2PD 2820108 Ki = 234 nM T08123 CRH5G3 5723593 Ki = 740 nM T08123 C85LJF 6463365 IC50 = 15.85 nM T08123 C02UYV 6918633 Ki = 5464 nM T08123 C0FV5J 7190424 IC50 = 215 nM T08123 C6XW2C 7190426 IC50 = 187 nM T08123 CPD45M 8272290 IC50 = 12000 nM T08123 CQ53PX 9567224 IC50 = 4100 nM T08123 CC90FJ 9869737 IC50 = 4600 nM T08123 C0BDP2 10313195 Ki = 2702 nM T08123 CSHT79 11056377 Ki = 240 nM T08123 C14SYJ 11088637 Ki = 2793 nM T08123 CFH5T7 11099263 Ki = 137 nM T08123 CQ29JI 11120348 Ki = 156 nM T08123 CID08M 16798824 IC50 = 200 nM T08123 CI5ST3 17982588 IC50 = 204 nM T08123 C5QWZ2 18561027 IC50 = 167 nM T08123 C5JWI9 21184460 Ki = 94 nM T08123 CR85BP 21184514 Ki = 863 nM T08123 C0ZGI1 21184532 Ki = 993 nM T08123 C8PBY4 21184553 Ki = 5583 nM T08123 CW1Q9P 21184562 Ki = 454 nM T08123 C19NOL 22500220 IC50 = 1500 nM T08123 C7YG1N 24759534 IC50 = 14 nM T08123 C7A5ET 24772735 Ki = 13 nM T08123 CJR3M7 25014542 IC50 = 15 nM T08123 CNQ9G5 25218180 IC50 = 46 nM T08123 C29RMK 36982503 IC50 = 12.59 nM T08123 CBY14D 39378356 IC50 = 48 nM T08123 CMI4D7 43668876 IC50 = 103 nM T08123 C8IHL7 44252884 IC50 = 1.3 nM T08123 C4X5CN 44444551 IC50 = 781 nM T08123 C7W5DZ 45790300 Ki = 2193 nM T08123 CB4JL5 45909952 IC50 > 10000 nM T08123 CVJU38 46233842 IC50 = 46 nM T08123 CQ9A7L 46234188 IC50 = 5 nM T08123 C0AF2X 46234666 IC50 = 2970 nM T08123 CPEO49 46843906 IC50 = 3.5 nM T08123 CGTM17 46898099 IC50 = 67 nM T08123 CM73EY 46912329 IC50 = 4900 nM T08123 C2B6VG 46912330 IC50 = 390 nM T08123 CXC70W 46912331 Ki = 182 nM T08123 C9MN1J 46912430 IC50 = 880 nM T08123 CQWY38 46912641 IC50 = 440 nM T08123 CZ3G6S 46913411 IC50 = 110 nM T08123 CV7T6O 47051749 IC50 = 343 nM T08123 CZ4MI0 49678035 IC50 = 351 nM T08123 C53SWY 49830719 IC50 = 22265 nM T08123 CYM4B1 49873378 IC50 > 1000 nM T08123 CAQ8F7 51356954 IC50 = 63.1 nM T08123 C5HP1Z 51356955 IC50 = 25.12 nM T08123 CJK6W0 51357233 IC50 = 19.95 nM T08123 CCP4R8 51357236 IC50 > 25118.86 nM T08123 CQ8O4Y 51357512 IC50 = 39.81 nM T08123 C90CUV 51357515 IC50 = 94 nM T08123 CIPU75 51357517 IC50 = 2511.89 nM T08123 CF1H2I 52109436 IC50 = 633 nM T08123 CCT8U0 54673065 IC50 = 770 nM T08123 C1ZF5H 54754832 Ki = 11 nM T08123 CK1Z7L 54755067 Ki = 7 nM T08123 CY9KA8 54755181 Ki = 13 nM T08123 CSY80Z 54755789 Ki = 9 nM T08123 CGAC06 56786904 IC50 = 1900 nM T08123 CCGZ21 56940771 Ki = 27 nM T08123 CDIS83 56940772 Ki = 4.2 nM T08123 CF5T4L 56941359 IC50 = 170 nM T08123 CJ7O0S 56941360 IC50 = 410 nM T08123 CZO64R 56941655 Ki = 2.4 nM T08123 CI92PK 56942076 Ki = 147 nM T08123 C6IQ2P 56943105 Ki = 0.3 nM T08123 CGA0P9 57334382 Ki = 776 nM T08123 C5TJ4U 57334383 Ki = 928 nM T08123 C5WX2V 57334384 Ki = 561 nM T08123 CQP86G 57334387 Ki = 341 nM T08123 CTF0M7 57334388 Ki = 64 nM T08123 CA95WC 57334531 Ki = 198 nM T08123 CQ0C7W 57334533 Ki = 53 nM T08123 CCE18Y 57334534 Ki = 293 nM T08123 CF46ZH 57334685 Ki = 4226 nM T08123 C0YD1F 57334686 Ki = 186 nM T08123 CO5I8C 57334687 Ki = 367 nM T08123 C2X1OV 57334689 Ki = 700 nM T08123 CZJM56 57334838 Ki = 286 nM T08123 CB0V4Q 57334992 Ki = 355 nM T08123 CN1C0Y 57334993 Ki = 348 nM T08123 CQVG63 57335145 Ki = 1598 nM T08123 C2YX3K 57335445 Ki = 2535 nM T08123 CVQO80 57335590 Ki = 2219 nM T08123 C9TB0Q 57336018 Ki = 143 nM T08123 CZ81QY 57336022 Ki = 1650 nM T08123 C1IX2E 57336023 Ki = 225 nM T08123 C4I0QW 58494270 Ki = 54 nM T08123 C2W0OD 58539094 Ki = 1 nM T08123 C5UTG9 58539095 Ki = 6 nM T08123 C7G2XB 58539106 Ki = 4 nM T08123 C60QVD 58539109 Ki = 2 nM T08123 C6CDB7 58539140 Ki = 1 nM T08123 CB3TQ8 58539146 Ki = 58 nM T08123 C8NG0L 58539237 Ki = 12 nM T08123 C19LBX 58539246 Ki = 3 nM T08123 C7WRQ5 58539268 Ki = 7 nM T08123 C97ZGJ 58539301 Ki = 3 nM T08123 CXJ63M 59603829 IC50 < 10 nM T08123 CQEU96 59603842 IC50 = 3.1 nM T08123 C9PUK6 59618824 Ki = 44 nM T08123 CPC0J1 59618832 IC50 = 530 nM T08123 C4NP7V 59618853 IC50 = 410 nM T08123 CPG7N9 59618867 IC50 = 830 nM T08123 CPKJ27 59618871 IC50 = 97 nM T08123 C30PWU 59618913 IC50 = 1600 nM T08123 CULS42 59618916 IC50 = 130 nM T08123 CQW85Z 59618941 IC50 = 390 nM T08123 C3NDI8 59618946 IC50 = 2400 nM T08123 CK08DV 59618947 IC50 = 68 nM T08123 C8OH4T 59618953 IC50 = 170 nM T08123 CZ6I4N 59618971 IC50 = 150 nM T08123 C0FJE7 59618977 IC50 = 3000 nM T08123 C1E5YI 59619022 IC50 = 86 nM T08123 C2IV1R 59619059 IC50 = 4700 nM T08123 CJXN91 59619097 IC50 = 300 nM T08123 C4EHP8 59619113 IC50 = 1900 nM T08123 CHMP08 59619145 IC50 = 250 nM T08123 CFW1M3 60196513 Ki = 301 nM T08123 C5FJU9 60197123 Ki = 160 nM T08123 C0PYI9 60197124 Ki = 97 nM T08123 CG0OM3 60197218 Ki = 189 nM T08123 C9MC6A 60197321 Ki = 133 nM T08123 CPG4K0 60197831 Ki = 2242 nM T08123 CSZ6I5 66556035 IC50 = 251.19 nM T08123 CWU8E6 66556279 IC50 <= 500 nM T08123 C7MD5X 66556536 IC50 = 1258.93 nM T08123 CD3WZ0 66827038 IC50 = 4 nM T08123 CUGS26 66828963 Ki = 44 nM T08123 C3AQY8 66829086 IC50 = 15 nM T08123 CSOR32 66829097 IC50 = 3 nM T08123 CN3WO7 66994399 IC50 = 6186 nM T08123 C4P2VS 67106997 IC50 = 7.943 nM T08123 CGD1O0 67107000 IC50 = 12.59 nM T08123 CC18RT 67107081 IC50 = 15.85 nM T08123 CH91GR 67107177 IC50 = 12.59 nM T08123 C9SV4B 67107224 IC50 = 19.95 nM T08123 CUF6E1 67107237 IC50 = 7.943 nM T08123 CJQ52M 67107333 IC50 = 10 nM T08123 CL7KA9 67107360 IC50 = 15.85 nM T08123 CIV97A 67107407 IC50 = 39.81 nM T08123 CMD36P 67108013 IC50 = 10 nM T08123 CV63UL 67240318 IC50 > 10000 nM T08123 CA4VO9 67814206 Ki = 5 nM T08123 CZ8U0Y 67817055 Ki = 9 nM T08123 C49CYH 67818467 Ki = 6 nM T08123 C2HYA3 67818622 Ki = 2 nM T08123 C59DOP 67988921 Ki = 6 nM T08123 C30CWB 68069662 Ki = 7.8 nM T08123 C6XF7V 68069685 IC50 = 11 nM T08123 CI9SU3 68069764 Ki = 4600 nM T08123 C2LFT7 68107702 IC50 = 39.81 nM T08123 C3KQW0 68107965 IC50 = 8.9 nM T08123 CP2Q3S 68108534 IC50 = 7.943 nM T08123 C6VMC2 68108924 IC50 = 63.1 nM T08123 C6QJH5 68239103 IC50 = 1231 nM T08123 CP61LD 68295403 Ki = 295 nM T08123 CQ1D0B 68778984 IC50 = 130 nM T08123 C5DGR9 69036886 IC50 = 167 nM T08123 C3C6EI 69048008 Ki = 557 nM T08123 CHF59A 69048861 Ki = 92 nM T08123 C7E1HF 69081779 IC50 = 140 nM T08123 CUG5E9 69081998 Ki = 2 nM T08123 CM38XA 69083959 IC50 = 99 nM T08123 CR05LF 69085771 Ki = 6 nM T08123 CQ86JW 69091994 Ki = 21 nM T08123 C72ZVX 69092378 Ki = 11 nM T08123 C5Y3OZ 69092949 Ki = 1 nM T08123 C4WG1A 69093006 Ki = 3 nM T08123 C0NA7R 69093113 Ki = 4 nM T08123 CN3A5C 69093123 Ki = 3 nM T08123 C8EF1H 69093313 Ki = 41 nM T08123 CER1B9 69093374 Ki = 0.7 nM T08123 C2U6AZ 69093445 IC50 = 36 nM T08123 C6Z9GS 69093717 Ki = 3 nM T08123 CJ91XV 69281457 Ki = 9 nM T08123 CK2PS4 69281523 Ki = 2 nM T08123 CNK07L 69281529 Ki = 6 nM T08123 CXKU75 69281543 Ki = 4 nM T08123 CV3XD9 69281569 Ki = 2 nM T08123 CN82OH 69281678 Ki = 8 nM T08123 CC9NG8 69281703 Ki = 2 nM T08123 CD07CR 69281708 Ki = 2 nM T08123 C3GTU1 69762142 IC50 > 10000 nM T08123 C9K3LU 69936228 IC50 = 251.19 nM T08123 CAVH70 69936275 IC50 = 125.89 nM T08123 CB3NM4 69936458 IC50 = 10 nM T08123 CR25CZ 69936757 IC50 = 199.53 nM T08123 CD0ME9 69936791 IC50 = 1258.93 nM T08123 CRO43B 69937003 IC50 = 7.943 nM T08123 CBO21X 69937058 IC50 = 50.12 nM T08123 C6Q7NH 70096101 Ki = 5 nM T08123 CJ96RN 70099013 Ki = 6 nM T08123 CC5Y7E 71060772 IC50 = 412 nM T08123 C48ZLN 71060894 IC50 = 10 nM T08123 C81ZNG 71060941 IC50 = 66 nM T08123 C10CHQ 71060955 IC50 = 15 nM T08123 CP4QU7 71060982 IC50 = 378 nM T08123 CGMJ84 71060999 IC50 = 17 nM T08123 CK35TB 71061025 IC50 = 5 nM T08123 C2UR3H 71061036 IC50 = 1 nM T08123 C94IAV 71061083 IC50 = 23 nM T08123 CT2N7Y 71061182 IC50 = 55 nM T08123 CI3LN8 71061196 IC50 = 12 nM T08123 CH0E6M 71061284 EC50 = 242 nM T08123 CY9E5Z 71061321 IC50 = 59 nM T08123 CTF14U 71061353 IC50 = 142 nM T08123 C8YF0R 71061365 IC50 = 17 nM T08123 CE31SP 71061394 IC50 = 49 nM T08123 CAOC46 71061450 IC50 = 145 nM T08123 CSZ1O5 71061479 IC50 = 56 nM T08123 CIZ49M 71061494 IC50 = 121 nM T08123 CWO0S3 71061505 IC50 = 7 nM T08123 C57NEV 71061537 IC50 = 9 nM T08123 CJ73DM 71154928 IC50 = 1.2 nM T08123 C0T8HO 71450027 Ki = 1 nM T08123 CJK05F 71451846 Ki = 2 nM T08123 CL0M4V 71451847 Ki = 1 nM T08123 CKW32R 71451848 Ki = 2 nM T08123 CH27NO 71451849 Ki = 3 nM T08123 C0DJ8P 71451850 Ki = 4 nM T08123 CVNI90 71453547 Ki = 10 nM T08123 CX4LE5 71453548 Ki = 6 nM T08123 CAN57Z 71455263 Ki = 20 nM T08123 C5R3PF 71455393 Ki = 7 nM T08123 CPY5K3 71457046 Ki = 33 nM T08123 C1X6YV 71457047 Ki = 20 nM T08123 CTA0O7 71457164 Ki = 1 nM T08123 CML7F1 71458913 Ki = 11 nM T08123 C56AHL 71460830 Ki = 8 nM T08123 CYR35K 71460831 Ki = 9 nM T08123 CR6O7Q 71462440 Ki = 7 nM T08123 C2BUG4 71519483 IC50 = 965 nM T08123 CBN10O 71531214 IC50 = 466 nM T08123 CDM85H 71531360 IC50 = 205 nM T08123 CBXY59 71548179 Ki = 0.5 nM T08123 CAO1X2 71553438 IC50 = 6 nM T08123 C7ZQI4 71553439 IC50 = 5 nM T08123 C4EG2A 71578245 IC50 = 23 nM T08123 CWNO83 71578246 IC50 = 47 nM T08123 C3HK8A 71578314 IC50 = 7270 nM T08123 CIH0S5 71578315 IC50 = 39 nM T08123 C5EQN0 71578667 IC50 = 1313 nM T08123 CDLM98 71578668 IC50 = 2168 nM T08123 C17PUR 71578669 IC50 = 76 nM T08123 CUJ0E2 71578670 IC50 = 13 nM T08123 CD1TB6 71578671 IC50 = 18 nM T08123 C2ARC8 71578672 IC50 = 1727 nM T08123 CU49PG 71578673 IC50 = 2112 nM T08123 CR86ZT 71578754 IC50 = 134 nM T08123 C52VUT 71578755 IC50 = 164 nM T08123 C8YW5N 71578756 IC50 = 211 nM T08123 C8UL0Q 71578757 IC50 = 253 nM T08123 C8F5ED 71578758 IC50 = 3305 nM T08123 C7WGE9 71578759 IC50 = 265 nM T08123 CE2OV5 71578843 IC50 = 179 nM T08123 C0MD7S 71578844 IC50 = 309 nM T08123 CB1M4Z 71578845 IC50 = 511 nM T08123 CZLQ18 71578846 IC50 = 2020 nM T08123 CH93UE 71578847 IC50 = 22128 nM T08123 C0R5BV 71578848 IC50 = 19542 nM T08123 C95CTL 71578849 IC50 = 2026 nM T08123 CM92KY 71578927 IC50 = 2470 nM T08123 CHV29Y 71578928 IC50 = 8 nM T08123 CZYD04 71578929 IC50 = 77 nM T08123 C1U9BV 71578930 IC50 = 26 nM T08123 CYS49J 71578931 IC50 = 75 nM T08123 C0QMZ1 71578932 IC50 = 67 nM T08123 C8IB6O 71578933 IC50 = 117 nM T08123 C87JUI 71579008 IC50 = 33 nM T08123 CAB95H 71579009 IC50 = 141 nM T08123 CZ0I3G 71579010 IC50 = 48 nM T08123 C8QZI2 71579011 IC50 = 581 nM T08123 CHGE58 71579086 IC50 = 3117 nM T08123 CR6GF2 71579087 IC50 = 162 nM T08123 CTW3D7 71579088 IC50 = 798 nM T08123 CD92LR 71579089 IC50 = 2068 nM T08123 C3NVQ1 71579090 IC50 > 4000 nM T08123 C20NET 71579091 IC50 > 100000 nM T08123 CA27BQ 71579092 IC50 > 100000 nM T08123 CEKJ06 71579169 IC50 > 100000 nM T08123 C9OJM2 71579170 IC50 = 4570 nM T08123 CGDW70 71579171 IC50 = 18000 nM T08123 C2T6XH 71579172 IC50 = 1230 nM T08123 CZW4T9 71579173 IC50 = 2270 nM T08123 C40ESW 71579260 IC50 = 9 nM T08123 C27CXJ 71579261 IC50 = 14 nM T08123 CW16ZS 71579330 IC50 = 16 nM T08123 CS7A4H 71579331 IC50 = 12 nM T08123 C1DSG0 71579332 IC50 = 28 nM T08123 CNTV53 71579333 IC50 = 48 nM T08123 C8YMF0 71579334 IC50 = 109 nM T08123 CS59YL 71579335 IC50 = 10 nM T08123 CGZ73I 71579413 IC50 = 14 nM T08123 C0YD6V 71579414 IC50 = 27 nM T08123 CBZ5H8 71579415 EC50 = 1599 nM T08123 CQ0KM2 71579416 IC50 = 281 nM T08123 CYA1G3 71579417 IC50 = 450 nM T08123 C5O6GN 71579418 IC50 = 498 nM T08123 CMO25Q 71579419 IC50 = 1177 nM T08123 CV65KO 71618473 EC50 = 62 nM T08123 C3OS8U 71714087 IC50 = 11 nM T08123 C92AZQ 71714088 IC50 = 14 nM T08123 CN1Y9I 71714230 IC50 = 7 nM T08123 CM6NE9 71714231 IC50 = 9 nM T08123 CG28AP 71714232 IC50 = 3 nM T08123 C91CRY 71714233 IC50 = 8 nM T08123 C67HDT 71714234 IC50 < 3 nM T08123 CRS05F 71714235 IC50 < 3 nM T08123 CVC19T 71714373 IC50 = 4 nM T08123 CD5C8J 71714374 IC50 = 4 nM T08123 C51ISR 71714375 IC50 = 31 nM T08123 C5HJK2 71714376 IC50 = 7 nM T08123 C70SJV 71714377 IC50 < 3 nM T08123 CK7T2U 71714378 IC50 = 150 nM T08123 CRA97Q 71716389 IC50 = 2512 nM T08123 CD6TF5 71717133 IC50 = 2020 nM T08123 CVN80C 71717134 EC50 = 435 nM T08123 C0YFP8 71718226 IC50 = 35 nM T08123 CM5SW1 71718384 IC50 = 55 nM T08123 CFSN02 71718965 IC50 = 88597 nM T08123 C8HMA7 71719424 IC50 = 168 nM T08123 CKNB62 71720020 IC50 = 9 nM T08123 C2BCG9 71720168 IC50 = 71 nM T08123 C27MEF 71720656 EC50 = 290 nM T08123 C8ON1P 71720813 EC50 = 731 nM T08123 C2JUF3 71720814 IC50 = 1747 nM T08123 CXH7N3 71736610 Ki = 1.2 nM T08123 C3UE2O 71736769 Ki = 3.1 nM T08123 C2OGC1 71736927 Ki = 4.1 nM T08123 CNU94W 71737255 Ki = 151 nM T08123 CIJ6V1 72191820 Ki = 0.7 nM T08123 CT9UK8 72201342 Ki = 3 nM T08123 C6T2UJ 72201343 Ki = 3 nM T08123 COGM19 72201489 Ki = 0.9 nM T08123 C6M1YO 72706006 IC50 = 20 nM T08123 CXP2V3 72706157 IC50 = 69 nM T08123 CYGI30 72706399 IC50 = 8 nM T08123 CA3E7M 72706402 IC50 = 20 nM T08123 C7A4BC 72706513 IC50 = 28 nM T08123 CCX6R1 72706517 IC50 = 9 nM T08123 C0XM9Z 72706586 IC50 = 8 nM T08123 C95GZV 72706839 IC50 = 26 nM T08123 CX48SV 72706841 IC50 = 5 nM T08123 C68GYC 72706904 IC50 = 122 nM T08123 CWN2A7 72706906 IC50 = 6 nM T08123 CLOE10 72706962 IC50 = 16 nM T08123 CCQ5I1 72707018 IC50 = 95 nM T08123 C3V8ZX 72707020 IC50 = 79 nM T08123 CX75YR 73352604 IC50 = 398.11 nM T08123 CHY9T6 76310861 Ki = 6 nM T08123 C4A0CF 76328935 Ki = 2 nM T08123 CAB9W0 76336221 IC50 = 53 nM T08123 C4Q5IN 76514427 Ki = 1640 nM T08123 C9WH0O 77068229 IC50 = 387 nM T08123 C8BAS5 77105954 IC50 = 710 nM T08123 C20QLI 77105957 IC50 = 390 nM T08123 CEOC93 77105960 IC50 = 540 nM T08123 C52TFP 77106161 IC50 = 280 nM T08123 C5RI9B 77106162 IC50 = 600 nM T08123 C12MFU 77106364 IC50 = 910 nM T08123 C4B3OS 77106759 IC50 = 160 nM T08123 C5NYW0 77106960 IC50 = 1300 nM T08123 CLB1A4 78319901 IC50 = 0.76 nM T08123 C0ED6J 78319902 IC50 = 2 nM T08123 CS9U2F 78321156 IC50 = 3.8 nM T08123 CUTK65 78321839 IC50 = 7.2 nM T08123 C9NL4K 78322146 IC50 = 41 nM T08123 CEF9C7 78323982 IC50 = 10 nM T08123 C6W5QH 78323983 IC50 = 2.2 nM T08123 CL06IB 85472082 IC50 = 15 nM T08123 C56VDQ 85472857 IC50 = 12 nM T08123 CY2PF9 85472971 IC50 = 98 nM T08123 CU6B5D 86275848 Ki = 0.06 nM T08123 CYD43G 86287677 IC50 = 108 nM T08123 CM2A5T 86287678 IC50 = 27 nM T08123 C4HZ0K 86287740 IC50 = 50 nM T08123 CN2H3I 86287744 Ki = 0.5 nM T08123 C0NT3J 86287745 IC50 = 85 nM T08123 CQ1OI2 86287807 Ki = 3 nM T08123 C7M1KT 86287812 Ki = 31 nM T08123 CNJO04 86287875 Ki = 4 nM T08123 CG9XP0 86287876 Ki = 6 nM T08123 CZ31RV 86295257 Ki = 3.5 nM T08123 C1HW4B 89735655 IC50 = 62 nM T08123 CKYX09 89887060 Ki = 46 nM T08123 C57VTG 89887105 Ki = 372 nM T08123 C67WIJ 89889447 Ki = 39 nM T08123 COLS74 89889448 IC50 = 31 nM T08123 CKB38T 89914324 IC50 = 20 nM T08123 CIA65G 89914405 IC50 = 42 nM T08123 C2J8EP 89914567 IC50 = 18 nM T08123 CJ8D0S 89914904 IC50 = 18 nM T08123 CEO2Z8 89915076 IC50 = 37 nM T08123 CZ75OC 89915123 IC50 = 5 nM T08123 CW8Z6M 90398640 IC50 = 134 nM T08123 CPN72Q 90400634 IC50 = 6.4 nM T08123 C0T1HM 90400705 IC50 = 4.4 nM T08123 CEU52A 90400735 IC50 = 2.6 nM T08123 CK1U9Q 90400782 IC50 = 0.8 nM T08123 CU83QB 90400825 IC50 = 13 nM T08123 CMR3Z2 90400868 IC50 = 83 nM T08123 CMXV30 90400979 IC50 = 0.7 nM T08123 CX59BA 90401078 IC50 < 0.6 nM T08123 CNT0B7 90401093 IC50 = 18 nM T08123 C7LN1D 91623338 IC50 = 204 nM T08123 CEPI85 102532139 IC50 = 30 nM T08123 C9JC0V 117653476 Ki = 23 nM T08123 C1TF9K 118368174 IC50 = 33 nM T08123 CJA6T0 118711382 IC50 = 496 nM T08123 CN26EQ 118711383 IC50 = 242 nM T08123 CKTW37 118711384 IC50 = 349 nM T08123 CN8R0C 118711385 IC50 = 880 nM T08123 C02PGS 118711386 IC50 = 66 nM T08123 CIZ89U 118711387 IC50 = 2290 nM T08123 C9YVC5 118711388 IC50 = 2489 nM T08123 CYZP82 118711389 IC50 = 12600 nM T08123 CP4I3E 118711390 IC50 = 32000 nM T08123 C2S3NT 118711391 IC50 = 4330 nM T08123 COJ9R7 118711392 IC50 = 91 nM T08123 CV8FB5 118711393 IC50 = 95 nM T08123 C3Q6ZG 118711394 IC50 = 2760 nM T08123 C38MFC 118711395 IC50 = 1260 nM T08123 CNX90H 118711396 IC50 = 1070 nM T08123 C2GXW0 118711397 IC50 = 2110 nM T08123 CYI4C5 118711398 IC50 = 2070 nM T08123 CBIA81 118711399 IC50 = 78 nM T08123 C4KEP1 118711400 IC50 = 373 nM T08123 C4EVI2 118711401 IC50 = 1350 nM T08123 C41FJN 118711402 IC50 = 12635 nM T08123 CJH46F 118711403 IC50 = 236 nM T08123 CUM9T7 118711404 IC50 = 549 nM T08123 C1V9IW 118711405 IC50 = 6202 nM T08123 CB5O6N 118711406 IC50 = 9124 nM T08123 CG40AO 118711407 IC50 = 1211 nM T08123 C06EWA 118711408 IC50 = 763 nM T08123 CE0W9G 118711409 IC50 = 21858 nM T08123 CNL54X 118711410 IC50 = 32000 nM T08123 CDTB86 118711411 IC50 = 32000 nM T08123 CJ03UP 118711412 IC50 = 1461 nM T08123 CW7VI0 118711413 IC50 = 400 nM T08123 CUV48F 118711414 IC50 = 488 nM T08123 CNV50B 118711415 IC50 = 525 nM T08123 CST6F7 118711416 IC50 = 5850 nM T08123 CZEO41 118711417 IC50 = 1145 nM T08123 CKUG73 118711418 IC50 = 115 nM T08123 C74FZL 118711419 IC50 = 110 nM T08123 CB47ZY 118714386 IC50 = 261 nM T08123 CP27FW 118714387 IC50 = 163 nM T08123 CN3X5T 118714393 IC50 = 31 nM T08123 C97GTN 118714394 IC50 > 10000 nM T08123 CQOY61 118714395 IC50 = 46 nM T08123 CS1F8A 118725474 IC50 = 115 nM T08123 CB8IJ7 118725475 IC50 = 5223 nM T08123 CIT2O4 118725476 IC50 = 393 nM T08123 CC8EJ6 118725477 IC50 = 117 nM T08123 CIQ5T2 118725478 IC50 = 80 nM T08123 CV8B3E 118725479 IC50 = 686 nM T08123 CT03NG 118725480 IC50 = 2243 nM T08123 CHJ78I 118725505 IC50 = 1199 nM T08123 CGJ75M 118725506 IC50 = 8 nM T08123 C5CY0G 118725507 IC50 = 111 nM T08123 CTR71E 118725508 IC50 = 2331 nM T08123 CZ7LM6 118725509 IC50 = 139 nM T08123 C54JEF 118725510 IC50 = 222 nM T08123 CR9ML7 118725554 IC50 = 99 nM T08123 CAD9B8 118731632 IC50 = 72 nM T08123 CBM50V 118731633 IC50 = 51.2 nM T08123 CJSX41 118731634 IC50 > 1000 nM T08123 CF8IT2 118731635 IC50 = 654 nM T08123 CE31VZ 118731636 IC50 > 1000 nM T08123 CPD5M4 118731637 IC50 > 1000 nM T08123 CSQ8D3 118731638 IC50 > 1000 nM T08123 C0HG6I 118731639 IC50 > 1000 nM T08123 C1QNH2 118731640 IC50 > 1000 nM T08123 CC4V7Z 118731641 IC50 > 1000 nM T08123 C84HRP 118731642 IC50 > 1000 nM T08123 CR0UN5 118731643 IC50 > 1000 nM T08123 C4WEK7 118731644 IC50 > 1000 nM T08123 CA04ZD 118731645 IC50 > 1000 nM T08123 CNEC23 118731646 IC50 > 1000 nM T08123 CNG07R 118731647 IC50 > 1000 nM T08123 C9J5VH 118731648 IC50 > 1000 nM T08123 C2YQK9 118731649 IC50 > 1000 nM T08123 CIU1F4 118731650 IC50 > 1000 nM T08123 C9ROB3 118731651 IC50 > 1000 nM T08123 CLOF30 118731652 IC50 > 1000 nM T08123 CM7RP3 118731653 IC50 > 1000 nM T08123 C0KM7P 118731654 IC50 > 1000 nM T08123 C2Y7MH 118733361 IC50 = 130 nM T08123 C39LIM 126691326 IC50 = 4.13 nM T08123 CYU38M 127046607 Ki = 305 nM T08123 CIA9X7 127047484 Ki = 159 nM T08123 COI8G1 127047659 Ki = 28 nM T08123 CO1SP2 127047756 Ki = 5610 nM T08123 C7BRS1 127048109 Ki = 30 nM T08123 CO8Z2N 129900111 IC50 = 714 nM T08123 CK8R5Y 134145931 IC50 = 130 nM T08123 CIP61L 134153498 IC50 = 754 nM T08123 C54FXD 134957362 IC50 > 10000 nM T08123 CA9ME4 135325094 IC50 = 5.55 nM T08123 CVSO41 135325140 IC50 = 6.39 nM T08123 CVN7D3 135399193 IC50 = 3830 nM T08123 CBV30L 135402333 IC50 = 3110 nM T08123 CMA49H 135406018 IC50 = 2170 nM T08123 C6NWV2 135438718 IC50 = 15400 nM T08123 CY06RE 135439090 IC50 = 110 nM T08123 CVQ6I5 135442567 IC50 = 2980 nM T08123 C0O2VG 135443554 Ki = 3450 nM T08123 CLIC03 135468562 IC50 = 13200 nM T08123 C1KLP4 135478724 IC50 = 3690 nM T08123 C2PRQ9 135481207 IC50 = 5400 nM T08123 C05WVF 135491980 IC50 = 20 nM T08123 CNU3X6 135541201 IC50 = 7270 nM T08123 C6DE1S 135543409 IC50 = 1700 nM T08123 C1DW2N 135553979 IC50 = 1340 nM T08123 CTM91E 135600848 IC50 = 2340 nM T08123 CRE6X9 135982538 Ki = 550 nM T08123 C3ZC0S 136035743 IC50 = 53 nM T08123 C9RT5K 136386182 IC50 = 280 nM T08123 C1ZNX7 136386185 IC50 = 1020 nM T08123 C2E4SY 136577433 IC50 = 1200 nM T08123 CK9V1P 137199823 IC50 = 10 nM T08123 CA1B4T 137631885 Ki = 136 nM T08123 CZ2WJ1 137632774 IC50 = 205 nM T08123 CT2BI3 137633878 IC50 = 9100 nM T08123 CJK0Y9 137635622 IC50 = 728 nM T08123 CE3TS9 137636366 IC50 = 2200 nM T08123 CS9H7X 137636896 IC50 = 102 nM T08123 C7XTV2 137637903 IC50 = 57000 nM T08123 C1D0ZQ 137639268 IC50 = 44 nM T08123 CKW84R 137641709 IC50 = 1995.26 nM T08123 COH0Z7 137642181 IC50 = 2900 nM T08123 CT76GD 137642252 IC50 = 15848.93 nM T08123 CLF8W2 137643090 IC50 = 64 nM T08123 C0PDY6 137643960 Ki = 23 nM T08123 CQTK16 137646685 IC50 = 256 nM T08123 C2WIN1 137647763 IC50 = 28 nM T08123 CO0G8M 137649243 IC50 > 25118.86 nM T08123 CH3CM6 137650444 Ki = 783 nM T08123 CTAP14 137651126 Ki = 95 nM T08123 CUY89G 137651440 IC50 = 210 nM T08123 CQY7I9 137651563 IC50 > 25118.86 nM T08123 CG6BX0 137653375 IC50 = 11000 nM T08123 C9XAD7 137653470 IC50 = 12000 nM T08123 C7EPY6 137654369 IC50 = 13000 nM T08123 C8VPB4 137654430 IC50 = 44 nM T08123 C1L0DX 137655129 Ki = 225 nM T08123 C12RCY 137657070 IC50 = 3600 nM T08123 CU3LS5 137657223 IC50 = 6700 nM T08123 C71WCI 137658381 IC50 = 6.6 nM T08123 CY1C7A 137658612 IC50 = 13000 nM T08123 CN2W4L 137659738 IC50 = 5800 nM T08123 CM9BJ8 137659810 IC50 = 93 nM T08123 C46OEV 137660994 IC50 = 170 nM T08123 CZ9BN4 138320062 IC50 = 0.001 nM T08123 C7HO6Z 138550167 IC50 = 2.6 nM T08123 C19EZB 138550184 IC50 = 20.2 nM T08123 CLXQ83 138550248 IC50 = 1 nM T08123 C3HO8V 138550388 IC50 = 4.4 nM T08123 CRS3P0 138550552 IC50 = 0.9 nM T08123 C3Z6KF 141301379 IC50 = 20 nM T08123 CQ9M7D 142423799 IC50 = 1530 nM T08123 CQJ1X6 142423813 IC50 = 0.94 nM T08123 CF8KR7 142423880 IC50 = 8.7 nM T08123 C3RWS0 145964556 IC50 = 130 nM T08123 CBKU04 145965102 IC50 = 5350 nM T08123 CV9GM5 145966574 IC50 = 6980 nM T08123 CE41QV 145971783 IC50 = 7490 nM T08123 C1S4OD 145972297 IC50 = 760 nM T08123 CK8P5F 145974450 IC50 = 550 nM T08123 CU3V0W 145975422 IC50 = 1500 nM T08123 CIYM29 145975752 IC50 = 5930 nM T08123 C85WPK 145976833 IC50 = 120 nM T08123 C5M4RL 145977765 IC50 = 490 nM T08123 COG17U 146405943 IC50 = 280 nM T08123 C9YT1C 146405944 IC50 = 160 nM T08123 CC84BD 146405947 IC50 = 370 nM T08123 CT1Q0U 146405949 IC50 = 370 nM T08123 CDX63Y 146405954 IC50 = 330 nM T08123 C4V1QD 146405955 IC50 = 370 nM T08123 CMEB27 146405958 IC50 = 980 nM T08123 CRO92Y 146405959 IC50 = 170 nM T08123 CDFY63 146405961 IC50 = 1120 nM T08123 CE8SG3 146405966 IC50 = 260 nM T08123 CNC6Y1 153407886 IC50 = 3.31 nM T08123 C2J7UI 154031581 IC50 = 3.21 nM T08123 CR2GM1 155511660 IC50 = 12.59 nM T08123 C0TSM8 155511739 IC50 = 19.95 nM T08123 C2MD1Q 155513187 IC50 > 10000 nM T08123 CNY51A 155514319 IC50 = 25.12 nM T08123 CU6QY4 155515764 IC50 > 10000 nM T08123 CN4IB6 155516354 IC50 = 19.95 nM T08123 C8G4EJ 155516586 IC50 = 39.81 nM T08123 CI8RQ9 155516974 IC50 = 2 nM T08123 C6H0FR 155517433 IC50 = 3.31 nM T08123 CSJY76 155517776 IC50 = 25.12 nM T08123 CVH0P8 155519454 IC50 = 19.95 nM T08123 CH60UK 155521075 IC50 = 12.59 nM T08123 CG20IT 155522201 IC50 > 10000 nM T08123 C9TSH7 155522966 IC50 = 31.62 nM T08123 CZY05O 155524160 IC50 = 25.7 nM T08123 CZW45D 155525803 IC50 = 39.81 nM T08123 CE9KC4 155529925 IC50 > 10000 nM T08123 C8P4QZ 155530738 IC50 = 12.59 nM T08123 CR70GX 155532115 IC50 = 25.12 nM T08123 C2CG1A 155537016 IC50 > 10000 nM T08123 CH3I8Z 155539469 IC50 = 10 nM T08123 CB0OK8 155540491 IC50 = 19.95 nM T08123 CL3MR0 155542649 IC50 = 50.12 nM T08123 CI84SJ 155543889 IC50 > 10000 nM T08123 CO1CN9 155547476 IC50 = 25.12 nM T08123 CV4B5R 155548069 IC50 = 15.85 nM T08123 CC1LI7 155550279 IC50 = 39.81 nM T08123 C93CKT 155553547 IC50 = 63.1 nM T08123 CX8GR9 155553934 IC50 = 15.85 nM T08123 CJ1BF3 155557829 IC50 = 1 nM T08123 C8HWI4 155558510 IC50 = 7.943 nM T08123 C4M9WK 155558971 IC50 = 9.73 nM T08123 CBO2R8 155561624 IC50 = 19.95 nM T08123 CM6L9J 155562224 IC50 = 12.59 nM T08123 CYQI51 155562763 Ki = 3900 nM T08123 C4BWO7 155566862 IC50 = 19.95 nM T08123 CS12BT 155569011 IC50 = 13 nM T08123 CP17HA 155569379 IC50 = 63.1 nM T08123 D01OXV 76328936 Ki = 2 nM T08123 D01XYD 16760524 IC50 = 22 nM T08123 D07ADX 54764565 IC50 = 11 nM T08123 D0B6KT 72706837 IC50 = 278 nM T08123 D0J5FK 58539171 Ki = 1 nM T08123 D0R2WK 16038120 IC50 = 6.1 nM T08123 D0U3NI 53246941 IC50 = 16 nM T08123 D0WK9R 72706840 IC50 = 3 nM T08123 D0YQ8V 46236221 IC50 = 35 nM T56588 D0I0DL 3689 IC50 = 75900 nM T56588 C63KYD 66637 EC50 = 10000 nM T56588 CD48TY 694463 IC50 = 426000 nM T56588 CD5RW2 1279398 IC50 = 1400 nM T56588 C5Z6NT 3113150 IC50 = 2700 nM T56588 CXF09D 4231127 EC50 = 2800 nM T56588 CN85UI 4235339 IC50 = 2700 nM T56588 CI28HT 22432385 EC50 = 6700 nM T56588 CA72VD 44322229 IC50 = 14000 nM T56588 CIC1G6 46861929 IC50 = 3900 nM T56588 C39CGI 56653056 IC50 = 50000 nM T56588 C4KWB0 56654447 EC50 = 29000 nM T56588 C7XPS1 66727815 IC50 = 2400 nM T56588 D06XGK 105074 EC50 = 78000 nM T56588 D09HXX 4787937 IC50 > 10000 nM T04123 CU5ND3 57514697 IC50 > 200000 nM T04123 C0IJ2X 118737463 IC50 > 50000 nM T04123 C12OHP 122187565 IC50 > 50000 nM T04123 CXHR32 122187566 IC50 > 50000 nM T04123 C59OUG 122187567 IC50 > 50000 nM T76285 C0NJ2B 645025 IC50 = 350 nM T76285 CRM9S6 674647 IC50 = 1150 nM T76285 CN06WE 685663 IC50 = 630 nM T76285 C5UAR2 910374 IC50 = 3220 nM T76285 C83UKT 1223927 IC50 = 5980 nM T76285 CAX45S 3332652 IC50 = 1810 nM T76285 CW7YG3 3724041 IC50 = 3420 nM T76285 C9KGH4 13224102 IC50 = 3150 nM T76285 CG19LI 23342610 IC50 = 1260 nM T76285 C7I0CN 32937631 IC50 = 2772 nM T76285 CRZ62F 73355036 IC50 = 1270 nM T76285 C5M9IT 101891745 Ki = 68100 nM T76285 C8HPR3 127045881 IC50 = 369 nM T76285 CZ58ER 127045883 IC50 = 856 nM T76285 CM1QX6 132584225 IC50 = 2250 nM T76285 CDF79W 145950387 IC50 > 100000 nM T76285 C9VIW7 145951405 IC50 = 1140 nM T76285 CI0DE8 145952129 IC50 > 100000 nM T76285 C8WY3S 145952263 IC50 > 100000 nM T76285 CCE24P 145953494 IC50 > 100000 nM T76285 CHSD24 145955401 IC50 > 100000 nM T76285 CVM5E8 145957948 IC50 > 100000 nM T76285 CVC6A1 145958826 IC50 > 100000 nM T76285 C8LWV3 145958854 IC50 = 390 nM T76285 CYG9B0 145958960 IC50 = 360 nM T76285 C6YJ4N 145961405 IC50 > 100000 nM T76285 CJ0IQ6 145962930 IC50 > 100000 nM T76285 CHN5E3 145974297 IC50 = 2420 nM T76285 CWKM51 145979441 IC50 = 230 nM T76285 CDQ0T6 145981705 IC50 = 410 nM T76285 CE8N3X 145987231 IC50 = 12400 nM T76285 C87AJL 145988932 IC50 = 1260 nM T76285 CVWI49 145990949 IC50 = 2260 nM T76285 CTQ21M 145991361 IC50 = 1220 nM T76285 CPI0F4 145992202 IC50 = 320 nM T76285 CFW27N 145992560 IC50 = 510 nM T76285 CI4C2R 145992946 IC50 = 2370 nM T76285 C4QID1 145993905 IC50 = 1530 nM T76285 C5JWS2 155512949 IC50 = 6602 nM T76285 C83ARF 155516516 IC50 = 3424 nM T76285 CD0Q7G 155516795 IC50 = 1810 nM T76285 CZ1I3O 155522133 IC50 = 255 nM T76285 CUH9K1 155527208 IC50 = 1624 nM T76285 C4HMC0 155530954 IC50 = 1079 nM T76285 CVX03O 155532639 IC50 = 1790 nM T76285 C0SBV5 155532733 IC50 = 1203 nM T76285 C64ULP 155536432 IC50 = 710 nM T76285 C1J0QI 155537162 IC50 = 1550 nM T76285 CE29XR 155538214 IC50 = 5426 nM T76285 CT98MF 155538277 IC50 = 807 nM T76285 CV3YF4 155540276 IC50 = 1525 nM T76285 CYH39A 155541761 IC50 = 2578 nM T76285 C10HXE 155543015 IC50 = 2409 nM T76285 CB8J0V 155549452 IC50 = 1014 nM T76285 CB2PX0 155549933 IC50 = 230 nM T76285 CI17FY 155556622 IC50 = 13520 nM T76285 CP6TE8 155557159 IC50 = 1510 nM T76285 C3RFG8 155559027 IC50 = 490 nM T76285 C1B4XC 155560220 IC50 = 1354 nM T76285 CV3X5K 155560593 IC50 = 3963 nM T76285 CGZ6L8 155561305 IC50 = 2675 nM T76285 CMNZ48 155561927 IC50 = 2892 nM T76285 C25AMC 155563065 IC50 = 214 nM T76285 CE1JW7 155564260 IC50 = 20510 nM T76285 C9XDT6 155566859 IC50 = 254 nM T76285 C75NHE 155567060 IC50 = 1724 nM T76285 C2UO0Y 155568526 IC50 = 1240 nM T76285 CTJK02 155568923 IC50 = 47010 nM T76285 CVTY16 155569460 IC50 = 2267 nM T60366 D0L4FS 5280961 IC50 = 26000 nM T60366 D0U3EP 445154 IC50 = 19000 nM T60366 CVIJ45 10520980 IC50 = 7400 nM T60366 CXVZ64 10542828 IC50 = 5200 nM T60366 CG1QD8 10689330 IC50 = 3900 nM T60366 CL79EJ 44418841 IC50 = 1.95 ug.mL-1 T60366 C15SEA 44418843 IC50 = 7.83 ug.mL-1 T60366 CM5X6O 44559035 IC50 > 30000 nM T60366 CXD56M 44559036 IC50 = 2200 nM T60366 CYP32C 44559037 IC50 = 2100 nM T60366 C4N6IJ 44559077 IC50 = 1100 nM T60366 CQZ5A3 44559078 IC50 = 2300 nM T60366 D04FIN 629965 IC50 = 3400 nM T60366 D04ZDD 44559034 IC50 = 2600 nM T60366 D0F3QP 5889042 IC50 = 4700 nM T60366 D0N4YR 10712965 IC50 = 3600 nM T16993 D0AF6O 71731823 IC50 = 3.3 nM T16993 D0OB0F 5328940 IC50 = 490 nM T16993 D06KTJ 53252276 IC50 = 51 nM T16993 D0E3TC 44259 IC50 = 1.8 nM T16993 D0T3ME 156422 IC50 = 17000 nM T16993 CB7WK3 5938113 IC50 = 42700 nM T16993 C5HW8Y 9949798 IC50 = 480 nM T16993 CACS26 11561968 Ki > 2000 nM T16993 CU0E8O 11690457 Ki > 2000 nM T16993 C3VRO9 44557921 IC50 > 10000 nM T16993 CLS29B 46872626 IC50 > 10000 nM T16993 CEQN27 52936621 Ki > 1000 nM T16993 C8NA4L 53384644 IC50 > 30000 nM T16993 C9UD0Y 56599956 IC50 = 25 nM T16993 C1MR8Q 60097495 IC50 > 1000 nM T16993 CV63UL 67240318 IC50 > 10000 nM T16993 CBE1V7 69284028 IC50 = 2.6 nM T16993 CPG3A5 86302574 IC50 > 30000 nM T16993 CE4GW0 123328993 IC50 = 210 nM T16993 C28QUP 137652864 IC50 = 5911 nM T16993 C38KLH 138393287 IC50 = 0.49 nM T16993 C2MD1Q 155513187 IC50 > 10000 nM T16993 C1RD6I 155520028 IC50 = 4.7 nM T16993 CWB35U 155523839 IC50 > 4000 nM T16993 CID82K 155524475 IC50 = 14 nM T16993 C4ZUI1 155524823 IC50 = 410 nM T16993 CLO7U1 155525161 IC50 > 4000 nM T16993 CNX69I 155525990 IC50 = 2.7 nM T16993 CMC65B 155527759 IC50 > 4000 nM T16993 C47UCR 155534288 IC50 = 57 nM T16993 C78MZC 155536330 IC50 = 2 nM T16993 CJ5FA1 155537070 IC50 > 1300 nM T16993 CO6CG8 155541167 IC50 = 510 nM T16993 CDG12I 155546428 IC50 = 440 nM T16993 CBO07E 155554038 IC50 = 460 nM T16993 CU8L9S 155554641 IC50 = 440 nM T16993 C3CSG4 155554781 IC50 = 10 nM T16993 CJQ65O 155560050 IC50 = 31 nM T16993 CP9HG1 155563860 IC50 > 4000 nM T16993 D09PTP 57325421 IC50 = 85 nM T16993 D0K5UF 72710568 IC50 = 2 nM T73475 D00MDP 466151 IC50 = 54 nM T73475 D05VZE 119031 IC50 = 4.1 nM T73475 D0MW3H 9824350 IC50 = 18.5 nM T73475 D0N4IV 10718956 IC50 > 1000 nM T73475 D0U2BH 65064 IC50 = 21500 nM T73475 D00UCC 9827497 IC50 = 11000 nM T73475 D01DVX 9847838 IC50 = 466 nM T73475 D03BOZ 3342298 IC50 = 210 nM T73475 D05VNG 9908389 IC50 = 11 nM T73475 D0P8YC 5362422 IC50 = 2.4 nM T73475 D0T9HG 132519 IC50 = 33 nM T73475 D0Y1XT 128564 IC50 = 30 nM T73475 CNA81R 1836 IC50 > 50000 nM T73475 CY78XM 4218 Ki = 30 nM T73475 CFY8Q2 4230 IC50 = 232 nM T73475 CDJS43 154136 IC50 = 460 nM T73475 C50IPY 154137 IC50 = 366 nM T73475 C7ROG5 177347 IC50 > 10000 nM T73475 C4U7SY 401129 IC50 = 72000 nM T73475 CV60YH 445010 IC50 = 3393 nM T73475 CK9M3P 445018 IC50 > 10000 nM T73475 C4D7TS 448002 Ki = 13000 nM T73475 CG1I8P 467296 IC50 > 100000 nM T73475 CTPW02 467297 IC50 > 100000 nM T73475 C9I8WB 478379 Ki = 3 nM T73475 CP0JM7 2109230 Ki = 10000 nM T73475 CN6E3U 2366268 IC50 > 10000 nM T73475 CY3TD6 3348132 Ki > 2000 nM T73475 CQ4VL5 5287415 IC50 = 3900 nM T73475 CJ3QI1 5288814 IC50 > 10000 nM T73475 C5IDT0 5289314 Ki = 850 nM T73475 CQEF36 6539670 IC50 = 180 nM T73475 CP7BG0 6852146 EC50 = 4 nM T73475 CN5L2B 6852147 IC50 = 460 nM T73475 C7Y1BX 9543420 IC50 = 886 nM T73475 CIXD67 9802768 IC50 > 10000 nM T73475 CQ46XD 9804842 IC50 = 20000 nM T73475 C6KJ9W 9822461 IC50 = 1700 nM T73475 C1MPW9 9823182 IC50 > 50000 nM T73475 C8IMT2 9847787 IC50 = 2.2 nM T73475 C7VXJ5 9848025 IC50 = 2.2 nM T73475 C4IEK0 9850035 IC50 = 9000 nM T73475 C8GE7U 9862764 IC50 > 50000 nM T73475 CJS23I 9868333 Ki = 25 nM T73475 CG17NZ 9869811 IC50 > 10000 nM T73475 C38BVX 9870100 IC50 > 1000 nM T73475 CHU9I8 9871883 IC50 = 7000 nM T73475 C0ZT7A 9883002 Ki = 96000 nM T73475 CZBK85 9886177 IC50 > 50000 nM T73475 C4PB5Z 9887544 IC50 = 3 nM T73475 C3ZG6O 9887870 IC50 = 7200 nM T73475 CD1U5P 9889190 IC50 > 10000 nM T73475 C27HMG 9889517 IC50 = 0.78 nM T73475 CH69LT 9892815 Ki = 7000 nM T73475 CSIB97 9896504 IC50 > 30000 nM T73475 C2R5CX 9905493 IC50 = 895 nM T73475 CN6WJ1 9909994 IC50 = 440 nM T73475 CM2F7R 9910302 IC50 = 1.2 nM T73475 CK5OV9 9930210 IC50 = 39 nM T73475 CDXR37 9933197 IC50 > 10000 nM T73475 C65ION 9935032 IC50 > 10000 nM T73475 CG38KL 9936728 Ki = 1.5 nM T73475 C16HTN 9948666 Ki = 3400 nM T73475 CN76XI 9957653 IC50 = 925 nM T73475 CVG0O2 9959014 IC50 > 1000 nM T73475 CFQ15E 9976696 IC50 = 45 nM T73475 C0HL2X 9976697 IC50 = 30 nM T73475 C09LSY 9979489 Ki > 6368 nM T73475 CO09PN 9983251 IC50 = 931 nM T73475 CJGR30 9983604 IC50 = 2590 nM T73475 CB2J3S 9999667 IC50 = 2000 nM T73475 C6U3CK 10006134 IC50 = 905 nM T73475 CR7T3J 10009978 Ki = 177 nM T73475 CJ6H8O 10019658 IC50 = 2027 nM T73475 C6WHU4 10023722 IC50 = 18 nM T73475 CJR59P 10031295 Ki > 6368 nM T73475 CLXN48 10047373 IC50 = 16500 nM T73475 CAN59F 10047708 IC50 = 1.6 nM T73475 CLZ87W 10051236 Ki = 635 nM T73475 CJK0R1 10074190 IC50 = 3307 nM T73475 C8AEK4 10093420 IC50 = 0.3 nM T73475 CA6X2Z 10095338 IC50 = 1.1 nM T73475 CMY3X2 10098158 IC50 = 3.1 nM T73475 C2XV5J 10098250 IC50 = 1020 nM T73475 C3V2HW 10099112 IC50 = 15000 nM T73475 C7A8MI 10120093 IC50 > 10000 nM T73475 CYU19P 10127901 Ki > 6370 nM T73475 CH0UW2 10129190 Ki > 6370 nM T73475 CUG62E 10155007 IC50 > 40000 nM T73475 CLQ89T 10155008 IC50 > 40000 nM T73475 CR5H6E 10163627 Ki = 5858 nM T73475 CZO5V4 10164317 IC50 = 20 nM T73475 CGB27E 10174981 Ki > 6370 nM T73475 CL47AR 10175070 Ki > 6370 nM T73475 C4ULO6 10175077 Ki > 6370 nM T73475 C84ZQD 10175219 Ki > 6370 nM T73475 CIT0H4 10175323 Ki > 6370 nM T73475 C95IGP 10175331 Ki > 6370 nM T73475 CT7U0M 10175426 Ki > 6370 nM T73475 CK0P3F 10186536 Ki = 4075 nM T73475 C51RPY 10195069 Ki > 6370 nM T73475 CCHX74 10195307 Ki > 6370 nM T73475 C94KHT 10195527 Ki > 6370 nM T73475 CDG35O 10196192 Ki > 6370 nM T73475 C4K1MJ 10208262 Ki = 3502 nM T73475 CG8FA4 10218128 Ki > 6370 nM T73475 C7Y2US 10218353 Ki > 6370 nM T73475 CV5X8A 10224181 IC50 > 30000 nM T73475 C7T0WH 10229644 IC50 = 8570 nM T73475 CO8M7Q 10239526 Ki > 6370 nM T73475 CEO4X5 10239762 Ki > 6370 nM T73475 CU7TQ3 10239803 Ki > 6370 nM T73475 CBM0Y4 10252411 Ki < 100 nM T73475 C2V4MP 10253549 IC50 = 3245 nM T73475 CB6SE4 10256227 IC50 = 40 nM T73475 C0CE3N 10269452 IC50 = 4800 nM T73475 C0QS9V 10269453 IC50 = 590 nM T73475 CR7JN6 10279317 Ki = 79 nM T73475 C3IG0K 10280852 IC50 > 10000 nM T73475 CR48SA 10289842 Ki > 6370 nM T73475 CO60CU 10290029 Ki > 6370 nM T73475 CE1KM9 10311498 Ki > 6370 nM T73475 CJ15OB 10311501 Ki > 6370 nM T73475 C5F0EV 10311947 Ki > 6370 nM T73475 C7G6QW 10312268 Ki > 6370 nM T73475 CQ5IT9 10312372 Ki > 6370 nM T73475 CIDW49 10319098 Ki > 6368 nM T73475 CG23FV 10320328 IC50 = 5400 nM T73475 CJWH74 10321975 Ki > 6368 nM T73475 CQH5D4 10324032 IC50 = 5.9 nM T73475 C94ANQ 10347529 IC50 = 845 nM T73475 C9FU5G 10362663 IC50 = 909 nM T73475 CH89GT 10365752 IC50 = 3.6 nM T73475 CI0T8K 10366352 Ki > 6368 nM T73475 C6WZ4F 10367355 IC50 = 2424 nM T73475 CFKA79 10395015 Ki = 834 nM T73475 CS32HR 10435935 IC50 = 1.5 nM T73475 C5WV1N 10439082 Ki = 1336 nM T73475 CA7DM9 10474389 IC50 = 500 nM T73475 CNQZ36 10483139 Ki > 10000 nM T73475 C9XC8Y 10493383 IC50 = 2100 nM T73475 C6KD0A 10498747 IC50 = 23 nM T73475 C36OMW 10502172 IC50 = 1400 nM T73475 C5V8HJ 10502382 IC50 < 24 nM T73475 CSN17G 10502708 IC50 = 4200 nM T73475 CBNM82 10503128 IC50 = 105 nM T73475 C9LJR5 10503737 IC50 = 54 nM T73475 C2C7TE 10504472 IC50 = 450 nM T73475 C6D7JF 10506147 IC50 = 36000 nM T73475 CBT12Q 10522080 IC50 = 1082 nM T73475 CC2F5Y 10522311 IC50 = 821 nM T73475 CZ36JW 10523383 IC50 = 16000 nM T73475 CQEH42 10524134 IC50 = 263 nM T73475 CYU87N 10524260 IC50 = 612 nM T73475 COT07L 10525329 IC50 = 14000 nM T73475 C61GSD 10525562 IC50 = 642 nM T73475 C14XUW 10526101 IC50 = 1522 nM T73475 CJK6G1 10526509 IC50 = 420 nM T73475 CWLD37 10526788 IC50 = 7100 nM T73475 CHS9Q5 10527785 IC50 > 10000 nM T73475 CJ0D7G 10528505 IC50 = 1018 nM T73475 CO2R0P 10544323 IC50 = 10000 nM T73475 C4PK0U 10549114 IC50 = 30 nM T73475 C4TA1K 10549256 IC50 = 60 nM T73475 CHCI01 10549577 IC50 = 620 nM T73475 C2HJ1U 10549764 IC50 = 1695 nM T73475 CRHP20 10550304 IC50 = 2173 nM T73475 C7WQ5Z 10550399 IC50 = 140 nM T73475 CNQ75F 10551139 IC50 = 6086 nM T73475 CCH0K3 10551483 IC50 = 908 nM T73475 C5UD0A 10551910 IC50 = 100000 nM T73475 CNE73L 10552476 IC50 = 3290 nM T73475 CI8XG0 10554869 IC50 = 6800 nM T73475 CT7O9M 10569678 IC50 = 4500 nM T73475 C8RWE4 10569743 IC50 = 31000 nM T73475 CE14GM 10570702 IC50 = 7200 nM T73475 CS9Y3Q 10573446 IC50 = 520 nM T73475 C61IUN 10574937 IC50 = 183 nM T73475 C9L5OM 10579282 IC50 = 123 nM T73475 CIUO27 10593253 IC50 = 2546 nM T73475 CUTS47 10594564 IC50 = 7000 nM T73475 CN4Y6H 10594565 IC50 = 19000 nM T73475 CYNC76 10596158 IC50 = 11000 nM T73475 C0R8ND 10599533 IC50 = 710 nM T73475 CQCW86 10599579 IC50 = 785 nM T73475 CW18QK 10599594 IC50 = 27 nM T73475 CR1JI4 10600645 IC50 = 3400 nM T73475 C6RH4O 10601640 IC50 = 1200 nM T73475 CG32FM 10613145 IC50 = 1200 nM T73475 CZD9B3 10617580 IC50 = 1102 nM T73475 CL02BO 10618584 IC50 = 4500 nM T73475 C0JGS3 10621776 IC50 > 10000 nM T73475 CL5QN9 10622296 IC50 = 710 nM T73475 CL62YC 10622822 IC50 = 354 nM T73475 CZJB31 10622970 IC50 = 2694 nM T73475 C98KGO 10625860 IC50 = 1134 nM T73475 CL43CO 10627365 IC50 = 716 nM T73475 C7KGM3 10642071 IC50 = 1058 nM T73475 CWRY91 10642128 IC50 = 537 nM T73475 CI2QB9 10642965 IC50 = 381 nM T73475 C2O1XM 10647817 IC50 = 1100 nM T73475 C5RWF4 10648802 IC50 = 1283 nM T73475 C27QHB 10663143 IC50 = 2390 nM T73475 CGSX70 10664302 IC50 = 1860 nM T73475 C97KZU 10665624 IC50 = 4800 nM T73475 CF0E6H 10668745 IC50 = 7900 nM T73475 C8HK0C 10669534 IC50 = 1460 nM T73475 CAI72H 10670246 IC50 = 4900 nM T73475 CY6QC1 10670819 IC50 = 2690 nM T73475 CPG5O2 10671155 IC50 = 416 nM T73475 C09LJR 10671827 IC50 = 401 nM T73475 CXTP56 10688727 IC50 = 82 nM T73475 C0OJ9C 10689683 IC50 = 2200 nM T73475 CSA80H 10692194 IC50 = 8700 nM T73475 CS5CL7 10692307 IC50 = 39 nM T73475 CR5KF8 10692994 IC50 = 100000 nM T73475 CDI12G 10693559 IC50 = 17 nM T73475 CB70DA 10693592 IC50 = 9800 nM T73475 CVML68 10693881 IC50 = 8500 nM T73475 CW6CF7 10696226 IC50 = 2700 nM T73475 C6MWX8 10696713 IC50 = 22050 nM T73475 C4IWF2 10714988 IC50 = 7400 nM T73475 CO9KV7 10715115 IC50 = 89 nM T73475 CE1D6G 10716217 IC50 < 100 nM T73475 C0ZX6T 10717308 IC50 = 3100 nM T73475 C7OSW8 10718200 IC50 = 610 nM T73475 CI64YZ 10718883 IC50 = 824 nM T73475 C35MRE 10719092 IC50 = 785 nM T73475 C51DZG 10737732 IC50 = 7500 nM T73475 C1LS5U 10738104 IC50 = 240 nM T73475 CL74TG 10738165 IC50 = 53 nM T73475 C76ANK 10739335 IC50 = 483 nM T73475 C0T2VK 10740460 IC50 = 787 nM T73475 CKJD45 10741133 IC50 = 78000 nM T73475 CL64BU 10741592 IC50 = 16 nM T73475 C4MQ8L 10742072 IC50 = 840 nM T73475 CHW23E 10742387 IC50 = 79 nM T73475 CCH94Q 10743507 IC50 = 1890 nM T73475 C9ILP3 10745718 IC50 = 15000 nM T73475 CE09PI 10757715 IC50 = 4300 nM T73475 C68THN 10763851 IC50 = 922 nM T73475 CAG53Y 10764489 IC50 = 509 nM T73475 C0ZJB9 10764600 IC50 = 27680 nM T73475 CJE76M 10764871 IC50 = 7400 nM T73475 CQ0KM4 10765140 IC50 = 790 nM T73475 C7Q2EM 10767236 IC50 = 3000 nM T73475 CLAP90 10785969 IC50 > 1000 nM T73475 C2FA7J 10787997 IC50 = 3500 nM T73475 C16XQR 10788211 IC50 = 1400 nM T73475 C0DFB9 10788617 IC50 = 170 nM T73475 CNAE08 10788733 IC50 = 2100 nM T73475 CKV2O8 10789493 IC50 = 483 nM T73475 CM74LH 10789594 IC50 > 1000 nM T73475 C45UGJ 10789671 IC50 = 850 nM T73475 C9NZ4W 10789711 IC50 = 502 nM T73475 CWCD73 10805054 IC50 = 12300 nM T73475 CN8I3Z 10808172 IC50 > 9994 nM T73475 CT1AI4 10810573 IC50 = 2700 nM T73475 CV3ZA5 10812444 IC50 = 4350 nM T73475 CZB7L2 10812929 IC50 < 100 nM T73475 C4TF0K 10813874 IC50 = 490 nM T73475 CCIL63 10813879 IC50 = 680 nM T73475 CS7BY4 10816934 IC50 = 8600 nM T73475 CX2E1C 10829071 IC50 = 313 nM T73475 C3AI5Z 10831752 IC50 = 22000 nM T73475 CLK9P7 10832592 IC50 = 12848 nM T73475 CF50HD 10832925 IC50 = 77000 nM T73475 C5OG4U 10833497 IC50 = 5600 nM T73475 C48PYQ 10836923 IC50 = 497 nM T73475 CH8OV4 10837276 IC50 = 110 nM T73475 CF40VH 10837557 IC50 = 1700 nM T73475 CY4J9A 10838149 IC50 = 2400 nM T73475 C3UCL2 10854279 IC50 = 1500 nM T73475 CAU0I3 10885834 IC50 = 3950 nM T73475 CXHA75 10928874 IC50 = 9870 nM T73475 CG2DK0 11016448 IC50 = 1740 nM T73475 CODQ51 11016616 IC50 = 3660 nM T73475 C9RU4I 11059620 IC50 = 5650 nM T73475 C1N5PT 11070986 IC50 = 4370 nM T73475 C18EIZ 11071831 IC50 = 2650 nM T73475 CY1SR9 11113744 IC50 > 10000 nM T73475 C2YBQ7 11134935 IC50 = 8510 nM T73475 C43ONW 11202395 Ki > 636 nM T73475 CO7T3M 11261246 IC50 > 10000 nM T73475 CP17ID 11284983 IC50 = 866 nM T73475 C1IW7N 11292680 IC50 > 1000 nM T73475 C8C5AV 11294179 Ki > 10000 nM T73475 CLH50U 11318841 IC50 = 458 nM T73475 C0XR3B 11330861 IC50 = 1640 nM T73475 CQH57S 11342435 IC50 = 1100 nM T73475 C9ABX8 11397130 Ki > 6368 nM T73475 COS67B 11456566 IC50 = 3010 nM T73475 CJ46KN 11508259 Ki = 9000 nM T73475 C5VUM2 11517085 Ki > 50000 nM T73475 CHV2G1 11575995 Ki > 10000000 nM T73475 CNY92D 11640694 Ki > 60000 nM T73475 CK9F4P 11673778 IC50 > 50000 nM T73475 C28WNK 11682752 Ki = 295000 nM T73475 C3U6ZR 11697504 Ki > 50000 nM T73475 C7CED0 11733417 IC50 > 10000 nM T73475 CO8QT0 11753905 Ki = 6 nM T73475 CKM6P2 11795228 IC50 = 15740 nM T73475 CCSD72 11795621 IC50 = 41 nM T73475 C47OIA 11797154 IC50 = 920 nM T73475 CJ4VL3 11797382 IC50 > 1000 nM T73475 CCD4W2 11797992 IC50 = 2093 nM T73475 CHQR96 11798386 IC50 = 1032 nM T73475 CQ9HE2 11811551 IC50 = 4240 nM T73475 CLW3F1 11812791 IC50 > 10000 nM T73475 C02BWA 11967143 Ki > 2000 nM T73475 CB80OT 12000718 IC50 > 20000 nM T73475 C43PJZ 12000720 IC50 > 20000 nM T73475 C1AJO7 13968141 IC50 > 300000 nM T73475 CA2H8V 14303060 IC50 = 4100 nM T73475 CGH19T 15296844 IC50 > 300000 nM T73475 CB3A4Z 15941413 Ki = 48500 nM T73475 CA40FE 15941550 Ki = 31000 nM T73475 CM3D1L 15941553 Ki = 39000 nM T73475 CQ0ZL7 15941677 Ki = 18000 nM T73475 C6R1LD 15985818 IC50 = 961 nM T73475 CQS0F5 16719301 IC50 > 10000 nM T73475 C75XDI 16730519 IC50 = 1700 nM T73475 C2W1VA 16739287 Ki > 6000 nM T73475 C3S2TQ 17754305 IC50 > 40000 nM T73475 CSY0N8 18394511 IC50 > 300000 nM T73475 CK8MP3 20620240 Ki = 8600 nM T73475 CPC4G6 20620273 Ki > 10000 nM T73475 CPK09X 20651316 IC50 = 23 nM T73475 CG1BD4 20689551 IC50 > 10000 nM T73475 CAS84B 22004289 Ki = 237 nM T73475 C1MCG7 22004293 Ki = 605 nM T73475 C36WFA 22096205 IC50 > 100000 nM T73475 CZT64B 22484431 Ki > 10000 nM T73475 CD3U8A 23627203 Ki > 2500 nM T73475 C3TWS6 24178109 Ki = 1600 nM T73475 C5M3YW 24799779 Ki = 110000 nM T73475 CFL04M 24881245 IC50 > 300000 nM T73475 CLIC14 24881246 IC50 > 300000 nM T73475 C4FI5C 24901479 IC50 = 71000 nM T73475 CAQ9Z1 25022681 Ki > 6368 nM T73475 CA86UE 25049752 Ki = 823 nM T73475 C82NLV 25049754 Ki = 3000 nM T73475 C6QFV4 25049756 Ki = 4000 nM T73475 CU6M9K 25060725 IC50 = 20000 nM T73475 CF7X2P 25060975 IC50 = 32000 nM T73475 CVR52U 25066764 IC50 > 22 nM T73475 CA5DJ4 25138228 Ki = 128000 nM T73475 CX6D9J 25138245 Ki > 3000 nM T73475 C7A6JQ 25138250 Ki = 33000 nM T73475 C6N7EQ 25138258 Ki = 1336 nM T73475 C7AD1J 25138259 Ki = 311 nM T73475 CJ9TQ2 25138260 Ki = 1527 nM T73475 CUT8I7 25138261 Ki = 2992 nM T73475 CBD9X6 25138262 Ki = 3311 nM T73475 C8LX1S 25138263 Ki = 1145 nM T73475 C3OV1L 25138264 Ki > 6368 nM T73475 C92WVM 25138265 Ki = 811 nM T73475 CMCS41 25138266 Ki > 6368 nM T73475 C1FJV5 25138267 Ki > 6368 nM T73475 C9N6WT 25138268 Ki > 6368 nM T73475 CF4QI1 25138269 Ki > 6368 nM T73475 C6P5UL 25138270 Ki > 6368 nM T73475 CQE0L7 25138271 Ki = 2647 nM T73475 C59XWU 25138272 Ki = 726 nM T73475 C1TNQ3 25141117 IC50 = 475 nM T73475 CR35QP 25144971 IC50 > 10000 nM T73475 C0Y5BC 25145683 IC50 > 2500 nM T73475 CHR2P1 25183768 Ki > 25000 nM T73475 C6AR8O 42623563 IC50 > 100000 nM T73475 CX0VP7 42623564 IC50 > 100000 nM T73475 CPO1Z3 44123600 IC50 = 3025 nM T73475 CCI64J 44224245 IC50 = 7830 nM T73475 CAR34Y 44263877 IC50 > 10000 nM T73475 CEV08N 44263913 IC50 = 737 nM T73475 C5ZI0X 44263926 IC50 = 88 nM T73475 CO3C1E 44263994 IC50 = 2780 nM T73475 C9XJ7U 44264020 IC50 = 10000 nM T73475 C6L0MJ 44264021 IC50 = 369 nM T73475 CJ1WE7 44264036 IC50 = 776 nM T73475 C50QFR 44264375 IC50 = 3460 nM T73475 C6YT3K 44280285 Ki = 1420 nM T73475 C8XUJ3 44280321 Ki = 3225 nM T73475 CC2O3U 44280323 Ki = 78 nM T73475 CM2TZ4 44280335 Ki = 114 nM T73475 CIE09F 44280336 Ki = 5 nM T73475 CA1V6Y 44280345 Ki = 18 nM T73475 CI9L2E 44280411 Ki > 620 nM T73475 C96NMF 44287796 IC50 = 70 nM T73475 CQ5IG7 44287805 IC50 = 33 nM T73475 CHOV34 44287806 IC50 = 50 nM T73475 CYAG29 44287899 IC50 = 2 nM T73475 CX5QB3 44287917 IC50 = 10 nM T73475 CCM31I 44288043 IC50 = 10 nM T73475 C1YT7H 44288071 IC50 = 10 nM T73475 CF2DZ9 44288091 IC50 = 3.1 nM T73475 CMY2N4 44288092 IC50 = 1 nM T73475 CCS20R 44288093 IC50 = 1 nM T73475 C2Y0PK 44302023 IC50 > 10000 nM T73475 C5S3UO 44302024 IC50 > 10000 nM T73475 C8ERW6 44302042 IC50 = 8540 nM T73475 CWB83G 44302076 IC50 = 5150 nM T73475 CY1J9U 44302096 IC50 = 9128 nM T73475 CW94ZQ 44302164 IC50 > 10000 nM T73475 CQ54PZ 44302166 IC50 = 500 nM T73475 C9U3XT 44302167 IC50 = 5000 nM T73475 C5X1WY 44302183 IC50 > 10000 nM T73475 C7G3BN 44302200 IC50 = 24061 nM T73475 C70QWV 44302327 IC50 = 40000 nM T73475 CZP20C 44302339 IC50 = 7069 nM T73475 CO73BW 44302357 IC50 > 10000 nM T73475 CNL4E2 44302361 IC50 = 20 nM T73475 CCW65Y 44302378 IC50 = 2000 nM T73475 CYG80V 44302385 IC50 = 10000 nM T73475 C7ZBR4 44302396 IC50 = 1000 nM T73475 C8S5WT 44302397 IC50 = 2000 nM T73475 CPC25G 44302409 IC50 = 7960 nM T73475 C4QL0I 44302411 IC50 = 3000 nM T73475 C4NDA2 44302416 IC50 = 20498 nM T73475 C24ZWF 44302429 IC50 > 10000 nM T73475 CYL71W 44302432 IC50 = 2000 nM T73475 C5H6OV 44302627 IC50 = 15147 nM T73475 C6QR7C 44302634 IC50 > 10000 nM T73475 CG8KJ0 44302661 IC50 = 5470 nM T73475 CX1M3Q 44302666 IC50 = 6340 nM T73475 C36CQP 44302952 IC50 = 4450 nM T73475 CLH14M 44305978 IC50 = 5.7 nM T73475 CZ49UN 44305988 IC50 = 2.6 nM T73475 C6I8JA 44306058 IC50 = 25 nM T73475 CB5EY3 44306200 IC50 = 4.2 nM T73475 C0YOH1 44306202 IC50 = 2.5 nM T73475 CMA39E 44306203 IC50 = 1.6 nM T73475 CL58OS 44306208 IC50 = 900 nM T73475 CAY2S4 44306209 IC50 = 110 nM T73475 C27NJX 44306277 IC50 = 180 nM T73475 C6O1AN 44306279 IC50 = 2.8 nM T73475 C89IQW 44318090 IC50 = 3640 nM T73475 CLQ23M 44321485 Ki = 210 nM T73475 CT0O7Y 44321602 Ki = 4 nM T73475 CV8T3N 44321783 Ki = 370 nM T73475 C4E8GU 44321802 Ki = 2100 nM T73475 C7Z4DQ 44321887 Ki = 117 nM T73475 CFJ20T 44321932 Ki = 605 nM T73475 CW9S1N 44321967 Ki = 1800 nM T73475 CI5X0G 44339523 IC50 = 4.2 nM T73475 CB9K8T 44339536 IC50 = 3.3 nM T73475 C2R3XN 44339554 IC50 = 13 nM T73475 C2CRY1 44339556 IC50 = 8.6 nM T73475 CTBU53 44339564 IC50 = 29 nM T73475 C58OSK 44339567 IC50 = 4.2 nM T73475 CX2KJ3 44339574 IC50 = 68 nM T73475 CEK3G0 44339588 IC50 = 5.7 nM T73475 C7ZR6H 44339589 IC50 = 220 nM T73475 C0WP9C 44339590 IC50 = 8 nM T73475 C5C2LI 44339654 IC50 = 4.3 nM T73475 C2SZB1 44342614 IC50 = 20 nM T73475 CQ60YD 44360219 IC50 = 330 nM T73475 CT4C6P 44360260 IC50 = 17651 nM T73475 CY5I3O 44360286 IC50 = 637 nM T73475 C40OCB 44360287 IC50 = 38 nM T73475 C3IW9L 44360784 IC50 = 18 nM T73475 CGQ92A 44364037 IC50 = 12040 nM T73475 CN4T7Q 44364119 IC50 = 21420 nM T73475 CH4TE7 44364121 IC50 = 7136 nM T73475 CPE91Y 44364122 IC50 = 10471.29 nM T73475 C1F8XN 44364249 IC50 = 3162.28 nM T73475 CWM47H 44364250 IC50 = 10690 nM T73475 C3TPO7 44364266 IC50 = 21380 nM T73475 C90CYD 44367175 IC50 = 5235 nM T73475 C2DV0R 44367276 IC50 = 294 nM T73475 C5BAW2 44367284 IC50 = 1792 nM T73475 C2YG5E 44367285 IC50 = 6724 nM T73475 CUDF82 44367309 IC50 = 2083 nM T73475 C3EV2A 44384940 IC50 > 50000 nM T73475 C0XE8K 44384941 IC50 > 50000 nM T73475 C3IJO9 44384994 IC50 > 50000 nM T73475 CWGQ46 44404503 IC50 = 534 nM T73475 CLXM58 44404504 IC50 = 1260 nM T73475 C1K3QM 44406655 IC50 = 200 nM T73475 C6YG5S 44406678 IC50 > 1000 nM T73475 CT5PC9 44422672 IC50 = 150 nM T73475 CS9D5U 44422720 IC50 = 450 nM T73475 CNWM05 44422723 IC50 = 2000 nM T73475 C58LAY 44422724 IC50 = 1400 nM T73475 CDQU41 44422736 IC50 = 20000 nM T73475 CVUB56 44422737 IC50 = 2900 nM T73475 CB8G2W 44422743 IC50 = 1100 nM T73475 CFX42T 44422744 IC50 = 50000 nM T73475 C9EL7F 44422749 IC50 = 130000 nM T73475 CJN1K9 44439853 Ki > 6370 nM T73475 CV58YW 44441018 Ki > 6368 nM T73475 CV85PN 44441019 Ki > 6368 nM T73475 C5O2WK 44441020 Ki > 6368 nM T73475 CU67WS 44441021 Ki > 6368 nM T73475 CXZ53B 44441022 Ki > 6368 nM T73475 C8S7UT 44441023 Ki > 6368 nM T73475 CT4PZ9 44441024 Ki > 6368 nM T73475 CU9GE6 44441025 Ki > 6368 nM T73475 CB2IT4 44441026 Ki > 6368 nM T73475 CN4X2F 44441027 Ki > 6368 nM T73475 CPF45Y 44441028 Ki > 6368 nM T73475 CAM23N 44441029 Ki > 6368 nM T73475 C23BPG 44441030 Ki = 5371 nM T73475 C5YMT6 44441031 Ki > 6368 nM T73475 C9A6GJ 44441032 Ki > 6368 nM T73475 CYSU19 44441033 Ki > 6368 nM T73475 C7T6EI 44445816 IC50 = 1819.7 nM T73475 CG9JS8 44445817 IC50 = 7585.78 nM T73475 CBX8S1 44445818 IC50 = 2570.4 nM T73475 CCYD65 44445819 IC50 = 1584.89 nM T73475 C3XG5N 44445820 IC50 = 2290.87 nM T73475 C58PEZ 44445821 IC50 = 9120.11 nM T73475 CRS83Q 44445822 IC50 = 309.03 nM T73475 CPO4U0 44445823 IC50 = 7413.1 nM T73475 CEQ8O0 44445824 IC50 = 851.14 nM T73475 CEOB52 44445825 IC50 = 446.68 nM T73475 CKEG37 44445826 IC50 = 2570.4 nM T73475 CHO12U 44445827 IC50 = 1000 nM T73475 C85EBJ 44445828 IC50 = 10964.78 nM T73475 CIJ70S 44445829 IC50 = 1202.26 nM T73475 COYD74 44445830 IC50 = 10964.78 nM T73475 CJ2BU5 44563487 IC50 = 6150 nM T73475 CHQG04 44576676 Ki = 10000 nM T73475 CR65DO 44576708 Ki = 1800 nM T73475 C9CB2Z 44576709 Ki = 602 nM T73475 C2QFY7 44576710 Ki = 625 nM T73475 C0BQV5 44576711 Ki = 5500 nM T73475 CU2IP7 44576753 Ki = 6600 nM T73475 C2QE3W 44576754 Ki = 6000 nM T73475 C8QHV1 44576806 Ki = 8600 nM T73475 C93LDF 44576807 Ki = 289 nM T73475 C9T2KO 44576808 Ki = 4800 nM T73475 C4RL6Y 44576809 Ki = 3000 nM T73475 CJ41MB 44576851 Ki = 7000 nM T73475 C9PUW2 44576877 Ki = 5000 nM T73475 C1F8WD 44576903 Ki = 3100 nM T73475 CTA01K 44576904 Ki = 2200 nM T73475 CK68GT 44580539 Ki = 75 nM T73475 CXIY57 44580801 Ki = 4617000 nM T73475 C0OA8Y 44580802 Ki > 10000000 nM T73475 CNC4D7 44581071 Ki = 1500000 nM T73475 CDF48U 44581111 Ki > 10000000 nM T73475 C56WVI 46184724 Ki = 6000 nM T73475 CL2U4Z 46829322 Ki = 1500 nM T73475 CH0Z1E 46844314 Ki > 40000 nM T73475 C20BTY 46856241 Ki = 3769 nM T73475 C5L8GF 46871738 IC50 > 10000 nM T73475 C0S9WB 46919610 Ki = 47000 nM T73475 C2S7PK 46942365 Ki = 2000 nM T73475 C7XW1Q 50907084 Ki = 344 nM T73475 C8RL5Q 50907292 Ki = 4000 nM T73475 CAS94N 51346773 Ki = 11000 nM T73475 CP65WT 51346774 Ki = 26000 nM T73475 C5OIA2 51346775 Ki = 35000 nM T73475 CU2SX3 51355576 Ki > 10000 nM T73475 CLA96C 53232689 Ki = 970 nM T73475 C3BGW0 53233015 Ki = 18100 nM T73475 CWH47R 53319228 Ki = 984 nM T73475 CI3WL5 53323418 Ki = 120000 nM T73475 C6Y2EV 53374826 IC50 > 100000 nM T73475 C3LF0P 54580544 Ki > 10000 nM T73475 CVO09J 54581546 Ki = 3000 nM T73475 CD09BZ 54582543 IC50 > 10000 nM T73475 CK52YD 54583511 Ki = 6000 nM T73475 CG37UX 54587429 Ki = 7100 nM T73475 CL9SC3 54587769 Ki = 13500 nM T73475 CHS01Z 54669766 Ki = 160000 nM T73475 C7E9SG 54757202 Ki = 116000 nM T73475 C62FZC 56835063 IC50 = 57700 nM T73475 C0L2TS 56835169 IC50 = 39000 nM T73475 CQU16V 57339411 Ki = 10700 nM T73475 C6LM3B 57339412 Ki = 7000 nM T73475 CWH7V8 57561293 IC50 > 40000 nM T73475 CY1N3J 57792153 IC50 = 1242 nM T73475 CCKD80 58307579 Ki > 25000 nM T73475 CMW3O0 71451330 Ki > 200 nM T73475 C9QS6E 71456659 Ki > 2000 nM T73475 C1U0FV 71601333 IC50 = 1150 nM T73475 C6KEH0 71680708 Ki > 25000 nM T73475 C7DMX5 71680709 Ki > 25000 nM T73475 CFPM82 71680710 Ki > 12000 nM T73475 C9ZOM7 71680866 Ki = 4000 nM T73475 CQ68LT 71680868 Ki > 100000 nM T73475 CFH2V0 71681183 Ki = 4100 nM T73475 CV3X1T 71682766 Ki > 20000 nM T73475 C5EAO8 71682767 Ki > 100000 nM T73475 C80EYX 71682913 Ki > 50000 nM T73475 C41BYG 71682915 Ki > 20000 nM T73475 C93XEI 71682916 Ki = 36000 nM T73475 CQ29PJ 71682917 Ki > 200000 nM T73475 CFWN65 71683062 Ki = 5700 nM T73475 C50SID 71817098 Ki = 18500 nM T73475 C38IDL 73345835 Ki = 11 nM T73475 CW01EA 73349535 IC50 > 100000 nM T73475 C8ROG3 73350414 Ki = 91 nM T73475 CF7AB2 73350415 Ki = 50 nM T73475 C2PFM4 73351930 Ki = 230 nM T73475 CI09CY 73354906 Ki = 12 nM T73475 C6H5TU 73354941 Ki = 6000 nM T73475 CGQ8F3 86287515 IC50 = 100000 nM T73475 CJ37XE 86287516 IC50 = 100000 nM T73475 COV8I9 86291010 IC50 = 1008 nM T73475 CRT54C 101910871 IC50 = 100000 nM T73475 CYA92R 130282633 IC50 = 180 nM T73475 CO3QE2 130282636 IC50 = 210 nM T73475 CTN42D 132941363 IC50 = 100000 nM T73475 C83FAY 134130294 Ki = 3760 nM T73475 CHV2U1 135438561 IC50 > 10000 nM T73475 CA5JR6 136054481 IC50 > 10000 nM T73475 CV47JN 136054485 IC50 > 10000 nM T73475 CZ48WO 136054487 IC50 > 10000 nM T73475 C8FGT0 136054495 IC50 > 10000 nM T73475 CG70BZ 136054516 IC50 = 30 nM T73475 CSM57W 136054520 IC50 = 2000 nM T73475 CXNG40 136118011 Ki = 1000 nM T73475 C1IOH9 136118012 Ki > 6368 nM T73475 CIEW62 136380958 IC50 = 1000 nM T73475 C9HS7J 137287436 IC50 = 7.3 nM T73475 C0I6RH 137632487 IC50 = 1102 nM T73475 CZ8H6N 137661550 IC50 = 100000 nM T73475 CZ25LW 155512044 IC50 = 100000 nM T73475 D02EFQ 10549609 IC50 = 11000 nM T73475 D03AMR 9849669 Ki = 660 nM T73475 D04GOO 10111838 IC50 > 100000 nM T73475 D04PAW 16216218 IC50 = 44000 nM T73475 D04VPH 45376872 IC50 > 22000 nM T73475 D06EHW 11625778 IC50 > 5000 nM T73475 D06HSC 136117931 IC50 = 15000 nM T73475 D07DRT 46175162 Ki = 3000 nM T73475 D07GEL 10344307 Ki = 0.8 nM T73475 D07SPC 24857837 Ki = 2800 nM T73475 D08ELY 9838786 IC50 = 1100 nM T73475 D09GIL 66160 IC50 > 50000 nM T73475 D09ZOA 25049753 Ki = 5000 nM T73475 D0A4TC 446504 IC50 = 106 nM T73475 D0B0UI 44428664 IC50 = 100000 nM T73475 D0B3UN 44580458 Ki = 626 nM T73475 D0BI8T 44288042 IC50 = 0.23 nM T73475 D0G3YZ 11391583 IC50 > 98000 nM T73475 D0H6CK 10160968 Ki = 18 nM T73475 D0K4TI 49292 IC50 > 50000 nM T73475 D0N6CD 10565532 IC50 = 290 nM T73475 D0N8YA 159596 IC50 > 100000 nM T73475 D0Q4TA 10044321 IC50 > 50000 nM T73475 D0Q9LC 44385624 IC50 > 50000 nM T73475 D0R2BO 194777 IC50 = 8.3 nM T73475 D0W2UK 6914621 Ki = 259 nM T73475 D0XK7G 10445302 Ki = 4000 nM T73475 D0Y5IQ 44255320 IC50 = 5000 nM T73475 D0Y7NV 2220392 IC50 > 50000 nM T03896 D09ZZW 503536 IC50 = 1500 nM T03896 C6IQV0 482174 IC50 = 5700 nM T03896 CY61LO 487910 IC50 = 1700 nM T03896 C6K5JV 487911 IC50 = 16000 nM T03896 C3J5VH 487912 IC50 = 1000 nM T03896 CZNK70 487918 IC50 = 330 nM T03896 CDN3F2 487919 IC50 = 1630 nM T03896 CT76XW 487920 IC50 = 2100 nM T03896 CVA82G 487921 IC50 = 460 nM T03896 CBR46W 487922 IC50 = 1400 nM T03896 CAJ64Q 490750 IC50 < 1000 nM T03896 CMO49H 491114 IC50 = 4300 nM T03896 COB17R 492544 IC50 > 50000 nM T03896 C68MZE 492548 IC50 > 100000 nM T03896 C4JO9E 492549 IC50 = 3280 nM T03896 C1JEY2 492550 IC50 = 300 nM T03896 CRML27 492552 IC50 = 380 nM T03896 C84QRW 493418 IC50 = 5700 nM T03896 CY1WF7 497453 IC50 = 3000 nM T03896 C43PXV 503499 IC50 = 2400 nM T03896 C2BSI5 503516 IC50 = 14000 nM T03896 CFRT87 503517 IC50 = 5400 nM T03896 C3JB0U 503520 IC50 = 13000 nM T03896 CA72XJ 503521 IC50 = 5200 nM T03896 CF14KO 503522 IC50 = 7400 nM T03896 CH18YP 503523 IC50 = 4600 nM T03896 CG6T1D 503524 IC50 = 4100 nM T03896 CLY7T8 503525 IC50 = 750 nM T03896 C37MIA 503526 IC50 = 1000 nM T03896 C8U2AD 503527 IC50 = 12000 nM T03896 CO6R4G 503528 IC50 = 2000 nM T03896 CHA5F8 503529 IC50 > 50000 nM T03896 C41DVG 503530 IC50 = 21000 nM T03896 C5XRJ6 503531 IC50 = 1200 nM T03896 CI1V6W 503532 IC50 > 50000 nM T03896 C84DXH 503533 IC50 = 1400 nM T03896 C7R3CM 503534 IC50 = 2000 nM T03896 CCMU16 503535 IC50 = 3000 nM T03896 C1E4IO 504181 IC50 = 2700 nM T03896 CEJ6U1 504182 IC50 = 1800 nM T03896 CZDS90 504183 IC50 = 1600 nM T03896 C04ONL 504184 IC50 = 2200 nM T03896 C65XPH 504185 IC50 = 11000 nM T03896 CRZN68 504186 IC50 = 42000 nM T03896 CK8CA2 504187 IC50 > 60000 nM T03896 C01MYV 504188 IC50 = 5800 nM T03896 C4C5WD 504189 IC50 = 4300 nM T03896 CIB52E 504190 IC50 = 230 nM T03896 CQ6L1G 504191 IC50 = 12000 nM T03896 C4CW5A 504192 IC50 > 60000 nM T03896 C09ACU 504193 IC50 > 60000 nM T03896 C7T0AD 504194 IC50 = 1300 nM T03896 C7VZY1 504195 IC50 > 60000 nM T03896 CU4EK0 504196 IC50 = 3600 nM T03896 COUS53 504197 IC50 = 5300 nM T03896 CTE3B4 504198 IC50 = 7700 nM T03896 CT81MP 504676 IC50 = 3500 nM T03896 C9FI5K 504680 IC50 = 10600 nM T03896 C8IFN4 504681 IC50 = 31000 nM T03896 CV6OY3 506523 IC50 = 1400 nM T03896 CQX7S4 506524 IC50 = 390 nM T03896 CXD73I 506525 IC50 = 1800 nM T03896 C6ANI5 506528 IC50 = 9000 nM T03896 CRU30I 507613 IC50 = 900 nM T03896 CI8SQ4 511361 IC50 > 50000 nM T03896 C02LPN 511362 IC50 = 30000 nM T03896 CJIW67 511363 IC50 = 13000 nM T03896 C3KG1M 511364 IC50 = 43000 nM T03896 CU85HK 511365 IC50 = 10700 nM T03896 C20EKN 511366 IC50 = 5900 nM T03896 C3FX8J 511367 IC50 = 31000 nM T03896 C4DEY1 511368 IC50 = 3700 nM T03896 CC2J9M 511369 IC50 = 5600 nM T03896 CIU5M2 511370 IC50 = 11000 nM T03896 C5CG4I 511371 IC50 = 5000 nM T03896 CTO87P 511372 IC50 = 2700 nM T03896 C5BJ6S 511373 IC50 = 26000 nM T03896 CDWB40 511374 IC50 = 15000 nM T03896 CDH29C 511375 IC50 = 31000 nM T03896 C8ZJD7 511376 IC50 = 31000 nM T03896 CJ56OH 513150 IC50 < 10000 nM T03896 C5BN4U 513891 IC50 = 12000 nM T03896 CVI54C 657065 IC50 = 1200 nM T03896 CUC54L 3008068 IC50 = 5000 nM T03896 CJ5NO6 3008069 IC50 = 34000 nM T03896 CQO9Y3 3008070 IC50 > 32000 nM T03896 CXM1K9 3008071 IC50 > 50000 nM T03896 CJ2NY3 3008418 IC50 = 20000 nM T03896 CIJ2T0 3008419 IC50 > 50000 nM T03896 CWD1X0 3008420 IC50 = 14000 nM T03896 C4K2JP 3008421 IC50 > 50000 nM T03896 CAN83S 3008422 IC50 = 13000 nM T03896 CMDQ27 4468931 IC50 = 1800 nM T03896 CK9WY1 5278824 IC50 = 100 nM T03896 C5MEQ4 5278825 IC50 = 110 nM T03896 C1F0AN 5278826 IC50 = 45 nM T03896 CV0O6S 5482516 IC50 = 15600 nM T03896 CEM30Z 5483089 IC50 = 8900 nM T03896 CJL21S 9853197 IC50 = 60 nM T03896 CJW4M9 9917616 IC50 = 11000 nM T03896 C39ZBC 10207572 IC50 = 30000 nM T03896 CGA86Z 10259200 IC50 = 12000 nM T03896 CJ46UK 10439772 IC50 = 420 nM T03896 COM8C5 21148125 IC50 = 16000 nM T03896 C1TW3V 22209806 IC50 > 50000 nM T03896 C8GVX3 22209808 IC50 > 50000 nM T03896 C6AS7E 22209811 IC50 = 3300 nM T03896 CLW13P 22209812 IC50 = 1700 nM T03896 C1TA6Z 22209813 IC50 = 440 nM T03896 CGUC83 22210989 IC50 = 58000 nM T03896 CV97ER 22210996 IC50 = 18000 nM T03896 C2BA1K 22211000 IC50 = 27000 nM T03896 C78AKX 22211010 IC50 > 100000 nM T03896 CL7M9B 22211011 IC50 = 32000 nM T03896 C1L8TE 22211012 IC50 = 18000 nM T03896 C0NYS5 22211016 IC50 = 50000 nM T03896 C67QJW 22211018 IC50 > 100000 nM T03896 CV9S2O 22211019 IC50 = 13000 nM T03896 C4UB6Q 22211020 IC50 = 14000 nM T03896 CBUV46 22211021 IC50 = 62000 nM T03896 CS9B7N 22211022 IC50 > 100000 nM T03896 CK81WO 25078062 IC50 = 3400 nM T03896 CYDW71 44268661 IC50 > 60000 nM T03896 C6S3AT 44268682 IC50 > 60000 nM T03896 CDJ0X4 44308299 IC50 > 100000 nM T03896 CIO1C2 44308345 IC50 > 100000 nM T03896 CX14BI 44308422 IC50 > 100000 nM T03896 CE3PS8 44308752 IC50 = 34000 nM T03896 CK2P5O 44375061 IC50 > 50000 nM T03896 C4CVW1 44375110 IC50 > 50000 nM T03896 C72KUL 44375154 IC50 = 9400 nM T03896 C1SBO9 44375192 IC50 > 50000 nM T03896 C42GUE 44375229 IC50 = 5300 nM T03896 CX76FI 44388198 IC50 = 350 nM T03896 CVW6O4 44399745 IC50 = 79432.82 nM T03896 CDRP83 44399750 IC50 = 50118.72 nM T03896 CW6NY8 44399751 IC50 = 5011.87 nM T03896 CM5W8Q 44399752 IC50 = 6309.57 nM T03896 C34WSP 44399753 IC50 = 10000 nM T03896 CE0T1O 44399754 IC50 = 1995.26 nM T03896 CT86CR 44399784 IC50 = 25118.86 nM T03896 C6GWS9 44399837 IC50 = 31622.78 nM T03896 C4AI1T 44399861 IC50 = 100000 nM T03896 CTX79F 44399866 IC50 = 25118.86 nM T03896 CP4KB7 44399867 IC50 = 794.33 nM T03896 C0WRU5 44399868 IC50 = 15848.93 nM T03896 C8JP2A 44399889 IC50 = 50118.72 nM T03896 CO4H3V 44399938 IC50 = 10000 nM T03896 CYH7F9 44399975 IC50 = 6309.57 nM T03896 CZRF38 44399976 IC50 = 6309.57 nM T03896 CATH48 44399977 IC50 = 6309.57 nM T03896 CL9NS3 44399978 IC50 > 199526.23 nM T03896 C9YO4K 44399979 IC50 > 199526.23 nM T03896 CX8M3O 44400003 IC50 = 39810.72 nM T03896 C4X1OG 44400004 IC50 = 19952.62 nM T03896 C5EV1S 44400005 IC50 = 158489.32 nM T03896 CFRU27 44400006 IC50 = 199526.23 nM T03896 C7FO3T 44400007 IC50 = 251188.64 nM T03896 CA6P2U 44400008 IC50 = 100000 nM T03896 CQP47M 44400009 IC50 = 7943.28 nM T03896 CCRB97 44400010 IC50 = 3981.07 nM T03896 CT40SR 44400033 IC50 = 31622.78 nM T03896 CA96HO 44400076 IC50 > 1000000 nM T03896 CX7O2Z 44400112 IC50 > 199526.23 nM T03896 C6Z5NC 44400113 IC50 > 199526.23 nM T03896 C6PCE5 44400114 IC50 = 31622.78 nM T03896 C95CRD 44400115 IC50 = 19952.62 nM T03896 CW5G3Z 73347065 IC50 > 50000 nM T03896 C6TNQ8 135412361 IC50 = 800 nM T03896 C53AWL 135434400 IC50 = 100 nM T96685 D04VIS 5318517 IC50 > 50000 nM T96685 D0X8ED 2327 IC50 = 5520 nM T96685 CHO1C9 57411333 IC50 = 790 nM T96685 CWDS87 57411452 IC50 = 50 nM T96685 C80DZY 57411679 IC50 = 10 nM T96685 CFK47B 67974063 IC50 = 2000 nM T96685 C2AZ4Y 67974101 IC50 > 400000 nM T96685 C5WEF0 67974104 IC50 = 25 nM T96685 C1TDA4 67974531 Ki = 2900 nM T96685 CKF7Q0 88537798 IC50 = 2000 nM T96685 C3RG6K 118714691 IC50 < 316.23 nM T96685 C1RE2H 127048545 IC50 = 3200 nM T96685 C49ZUL 127048546 IC50 = 790 nM T96685 CMI9A1 127048547 IC50 = 16000 nM T96685 CZ0C2N 127049887 IC50 = 630 nM T96685 C1JKC3 127049888 IC50 = 40 nM T96685 C13CQL 127049889 IC50 = 130 nM T96685 C27EYZ 127050129 IC50 = 16000 nM T96685 CJY3X7 127050185 IC50 = 25 nM T96685 CUR27K 127050186 IC50 = 7.9 nM T96685 C2ZQ3K 127050187 IC50 = 50 nM T96685 CU25TE 127050188 IC50 = 130 nM T96685 CZ5HL0 127051361 IC50 = 100 nM T96685 CO9FC4 127051362 IC50 = 130 nM T96685 C6OQG1 127052625 IC50 > 400000 nM T96685 CGV38D 127052626 IC50 = 100 nM T96685 CID97C 127052627 IC50 = 320 nM T96685 C16QBR 127052916 IC50 = 25 nM T96685 CEN92U 139053061 IC50 = 9800 nM T96685 C30ADT 145720921 IC50 = 34600 nM T96685 C3Z7VP 145720922 IC50 = 31200 nM T96685 C2P8OS 155511240 IC50 > 50000 nM T96685 CC8BF7 155512761 IC50 > 50000 nM T96685 CH5Q6L 155513950 IC50 = 26080 nM T96685 CG5PJ1 155514298 IC50 > 50000 nM T96685 C8VIL0 155514673 IC50 > 50000 nM T96685 CO4UH6 155514972 IC50 > 50000 nM T96685 CL97GC 155519990 IC50 > 50000 nM T96685 CN5UZ3 155522384 IC50 > 50000 nM T96685 C5LD2B 155526242 IC50 > 50000 nM T96685 C83ERS 155527164 IC50 > 50000 nM T96685 CHD3X6 155531906 IC50 = 9360 nM T96685 CV94KJ 155536434 IC50 > 50000 nM T96685 CXRM78 155537131 IC50 = 4800 nM T96685 C4E3TM 155538663 IC50 > 50000 nM T96685 CRS3E7 155546305 IC50 > 50000 nM T96685 C9XI0U 155558113 IC50 > 50000 nM T96685 CV5R2F 155560152 IC50 > 50000 nM T96685 C9WB1Q 155563330 IC50 > 50000 nM T96685 CW4YG8 155565340 IC50 > 50000 nM T96685 C0S5VT 155569173 IC50 > 50000 nM T22976 D03TGJ 5282192 Ki = 10400 nM T22976 D07XSN 6253 IC50 > 1000000 nM T22976 CP25DX 65049 IC50 = 285000 nM T22976 CPJ56E 452395 IC50 = 1300 nM T22976 CUW3B2 491807 IC50 = 27000 nM T22976 C8WS5I 491808 IC50 > 1000000 nM T22976 CYTV93 491811 IC50 = 801000 nM T22976 CA89BP 6476766 IC50 = 6300 nM T22976 CJB97H 6476767 IC50 = 402000 nM T22976 CZ1A0R 10097595 IC50 = 6800 nM T22976 C0PHT1 14606828 IC50 = 320 nM T22976 C3KA2N 16098860 IC50 = 45000 nM T22976 CH5P6G 16098865 IC50 = 5200 nM T22976 CH04XP 16098866 IC50 = 2400 nM T22976 C8MT2I 16098867 IC50 = 23000 nM T22976 CLIM56 16098869 IC50 = 114000 nM T22976 CL3T9X 16098872 IC50 = 1900 nM T22976 CF47QA 16098873 IC50 = 45000 nM T22976 C5GB9K 16098879 IC50 = 1900 nM T22976 CI4T9J 16098880 IC50 = 23000 nM T22976 CAF50V 16098881 IC50 = 1800 nM T22976 CI78AT 16121720 Ki = 290 nM T22976 C4MUA1 22489180 IC50 = 801000 nM T22976 C68QKG 44418800 IC50 = 390 nM T22976 CQY8X5 44437450 IC50 = 120000 nM T22976 C5H7LS 44437451 IC50 = 28000 nM T22976 CD0AN5 44437452 IC50 > 500000 nM T22976 C4YH3T 44437453 IC50 = 120000 nM T22976 C9LD5Y 44437454 IC50 > 1000000 nM T22976 CMB67C 44437455 IC50 = 480000 nM T22976 C5QFP6 44437456 IC50 = 74000 nM T22976 CJO51G 44437457 IC50 = 44000 nM T22976 CE1I4N 44437473 IC50 = 55000 nM T22976 CC0I1J 44437474 IC50 = 61000 nM T22976 C08ZMK 44437475 IC50 = 6400 nM T22976 CNPK62 44437476 IC50 = 3800 nM T22976 C2QO0P 44437477 IC50 = 187000 nM T22976 C9OE0G 44437478 IC50 > 500000 nM T22976 CO0N8X 44437480 IC50 > 1000000 nM T22976 C3BJE2 46197226 IC50 > 500000 nM T22976 C8WR4I 46197456 IC50 = 250 nM T22976 C2Y0QN 46197457 Ki = 12 nM T22976 CPA6D7 46700799 IC50 = 230 nM T22976 CWJY16 46874452 IC50 = 43000 nM T22976 C1PCR5 46884564 IC50 = 46 nM T22976 C4NK8W 46884565 IC50 = 42 nM T22976 C48RWL 46884566 IC50 = 1100 nM T22976 CN9RI6 46884567 IC50 = 4000 nM T22976 CZX1E7 46885197 Ki = 150 nM T22976 C5EPV6 46885249 IC50 = 400 nM T22976 C8DP0M 46885250 IC50 = 150 nM T22976 CQWV32 46885301 IC50 = 300 nM T22976 CG74UX 46885302 IC50 = 150 nM T22976 CUR4G7 46913823 IC50 = 91 ug.mL-1 T22976 CSQL06 54768280 IC50 = 60 ug.mL-1 T22976 CB9DU0 54768281 IC50 > 200 ug.mL-1 T22976 CUN04G 54768283 IC50 > 200 ug.mL-1 T22976 C2P3CT 90663608 IC50 > 1000000 nM T22976 CV0HE2 135499520 IC50 > 500000 nM T22976 C4K1FL 136118006 IC50 > 500000 nM T22976 CQGF80 136118007 IC50 > 500000 nM T22976 CR37CF 136118008 IC50 > 500000 nM T22976 D00KWL 16098859 IC50 = 2500 nM T22976 D02CCD 44418795 IC50 = 500 nM T22976 D07GKK 16098875 IC50 = 9700 nM T22976 D0C7YS 160155 Ki = 20000 nM T22976 D0I6UV 6477686 Ki = 500 nM T22976 D0O7GD 452142 IC50 = 4700 nM T22976 D0W8AD 16098874 IC50 = 4700 nM T32590 D09KTS 24821094 IC50 = 2.89 nM T32590 D0E6XR 3062316 IC50 = 0.3 nM T32590 D0OB0F 5328940 IC50 = 40 nM T32590 D02TUL 118115473 Ki = 131 nM T32590 D08AOZ 86582336 IC50 = 28 nM T32590 D0E3TC 44259 IC50 = 21.6 nM T32590 D0G5XV 135565884 IC50 = 2.95 nM T32590 CK5N6B 23657635 IC50 = 28 nM T32590 CSNC57 25110758 IC50 = 560 nM T32590 C0GOX5 25110759 IC50 = 500 nM T32590 CC2R7S 25110760 IC50 = 310 nM T32590 C36FXD 25138012 IC50 = 2 nM T32590 CP6N4G 25138050 IC50 = 220 nM T32590 CJL25F 25169253 IC50 = 700 nM T32590 CA98KR 44432441 IC50 = 1400 nM T32590 C8ZRE3 53356518 IC50 = 55 nM T32590 CJBL48 56925034 IC50 = 119 nM T32590 CZ3TG1 59375154 IC50 = 172 nM T32590 CV63UL 67240318 IC50 > 10000 nM T32590 C7VJ6A 70647728 IC50 = 180 nM T32590 COU73Y 71226944 IC50 = 45 nM T32590 C40JOZ 71235465 IC50 = 256 nM T32590 C54XWG 72190869 IC50 > 10000 nM T32590 CX75YR 73352604 IC50 = 79.43 nM T32590 C64SIO 92042864 IC50 = 36 nM T32590 C8HYU9 117926195 IC50 > 10000 nM T32590 C37DUM 121293882 IC50 = 26 nM T32590 CXQR89 121294143 IC50 = 2.3 nM T32590 CFKD32 122191637 IC50 = 95 nM T32590 CV89JM 132231876 IC50 = 15 nM T32590 C59HOQ 134277578 IC50 = 0.55 nM T32590 C0PZ5R 134277599 IC50 = 0.67 nM T32590 C7PWJ2 134277617 IC50 = 0.14 nM T32590 CRA2H1 134277633 IC50 = 0.47 nM T32590 CXJ8I0 134277643 IC50 = 0.18 nM T32590 C02RIA 134277647 IC50 = 0.2 nM T32590 CGH42R 134277652 IC50 = 0.25 nM T32590 COA14U 134277654 IC50 = 0.18 nM T32590 CQK0B5 134277685 IC50 = 0.76 nM T32590 C6S8VC 134277696 IC50 = 0.32 nM T32590 C49PIO 134277748 IC50 = 0.39 nM T32590 CD7VK4 134277767 IC50 = 0.59 nM T32590 CZ5E6L 134277773 IC50 = 0.42 nM T32590 C2CFK7 134277780 IC50 = 0.29 nM T32590 C6E7LW 134277790 IC50 = 0.21 nM T32590 C6T7NW 134277796 IC50 = 0.16 nM T32590 CU8ZP5 134277800 IC50 = 0.22 nM T32590 CTR4K6 134277828 IC50 = 0.14 nM T32590 CJ03PU 135566610 IC50 = 55.7 nM T32590 CQ9A5I 135566611 IC50 = 241.4 nM T32590 C42TOW 135566612 IC50 = 77.5 nM T32590 CN48IF 135566613 IC50 = 440.9 nM T32590 C67IYS 135566618 IC50 = 73.8 nM T32590 CP5SD0 136016241 IC50 = 66.5 nM T32590 C3Z4AT 137321159 IC50 > 10000 nM T32590 CZOD53 137633880 IC50 = 132 nM T32590 C7BJY5 137636807 IC50 = 282 nM T32590 CO89DX 137649100 IC50 = 231 nM T32590 CINE03 137652514 IC50 = 464 nM T32590 C28QUP 137652864 IC50 = 883 nM T32590 C4OD9Q 145967187 IC50 = 2.5 nM T32590 CE31VG 145979714 IC50 > 10000 nM T32590 C9BX4U 145988956 IC50 = 2990 nM T32590 C2MD1Q 155513187 IC50 > 10000 nM T32590 C3NA2I 155519537 IC50 = 358 nM T32590 D01RHR 71519693 IC50 = 1.9 nM T32590 D04PEI 11467730 IC50 = 11000 nM T32590 D04TLI 23657507 IC50 = 0.4 nM T32590 D06BJG 71556703 IC50 = 1.4 nM T62820 D00ENY 33032 EC50 = 290 nM T62820 D03FZT 25195461 EC50 = 65 nM T62820 D0B6RA 9834591 EC50 = 23.4 nM T62820 D0T3DG 9886034 Ki = 2.2 nM T62820 D01VZE 67705089 Ki = 7.43 nM T62820 D0D4OW 57338826 Ki = 20.1 nM T62820 D01FUB 25125217 EC50 = 195 nM T62820 D0P4BQ 9857256 Ki > 10000 nM T62820 D0U5CS 213056 EC50 = 5.1 nM T62820 D0ZV0R 16660135 IC50 > 10000 nM T62820 C0MLE4 1217 Ki > 1000000 nM T62820 CL8RX5 1222 Ki = 51000 nM T62820 COM10L 1297 Ki = 20000 nM T62820 CSM0F5 5115 IC50 = 577000 nM T62820 CZBT42 73537 EC50 = 110000 nM T62820 C8NO0Z 77937 EC50 > 1000000 nM T62820 C9H6OS 92136 EC50 = 35000 nM T62820 CUBH61 101122 EC50 > 1000000 nM T62820 CP05EH 136950 EC50 = 3500 nM T62820 CLMU31 165627 EC50 > 1000000 nM T62820 C34YGT 173564 EC50 > 1000000 nM T62820 CUT07K 177491 Ki > 300000 nM T62820 CR68YU 231345 EC50 > 1000000 nM T62820 C37ROZ 439282 Ki = 230 nM T62820 CO9KU6 443586 Ki > 1000000 nM T62820 C0S8TR 521212 EC50 = 3000 nM T62820 C3EP1R 627502 EC50 = 360 nM T62820 CW0CU9 798232 EC50 = 794.33 nM T62820 CB6X3Q 851990 EC50 = 5011.87 nM T62820 CNI89V 1617110 Ki = 205000 nM T62820 C5F8YH 2733519 EC50 > 600000 nM T62820 CZV0P5 3246152 Ki = 2000 nM T62820 C0HCI6 3461070 EC50 = 15848.93 nM T62820 COJV81 4521898 EC50 > 10000 nM T62820 CZ1Q5P 4694355 Ki = 30000 nM T62820 C05WNA 5310956 EC50 = 380 nM T62820 C7J6KQ 6604704 EC50 = 13000 nM T62820 C9INH1 6604707 EC50 > 1000000 nM T62820 CD68LI 6604795 Ki > 1000000 nM T62820 C6QSA9 7157252 EC50 > 300000 nM T62820 CL2OR7 7504549 EC50 = 155 nM T62820 C9PJQ1 9794208 EC50 = 0.16 nM T62820 CL8JI1 9837114 EC50 = 37000 nM T62820 CG3EN9 9885546 Ki = 85 nM T62820 C31YKH 9885608 EC50 = 1500 nM T62820 C9ACB3 9979770 EC50 = 229 nM T62820 CH54PF 9991661 EC50 = 122000 nM T62820 C9HD5C 9999945 EC50 = 3365 nM T62820 C1LK5F 10002415 EC50 = 2013 nM T62820 C0GN6F 10012356 Ki > 1000000 nM T62820 CQJP31 10012681 Ki = 122000 nM T62820 C82AGD 10026879 EC50 = 421 nM T62820 C6T7VH 10050046 EC50 = 1041 nM T62820 CAU7N4 10059959 EC50 > 300000 nM T62820 CYD93S 10070087 EC50 = 939 nM T62820 CYZ69A 10089411 Ki = 2700 nM T62820 CH6LU7 10103891 EC50 > 1000000 nM T62820 C8H3UO 10176324 EC50 > 10 nM T62820 C9XQK6 10198133 EC50 = 3.9 nM T62820 CL4NP9 10198359 EC50 = 10000 nM T62820 CAZ8P0 10198574 EC50 > 300000 nM T62820 CFDX64 10241509 EC50 > 300000 nM T62820 C7DU2G 10249222 EC50 = 72 nM T62820 C3TAF8 10251009 EC50 = 304 nM T62820 CUA94S 10262421 EC50 > 300000 nM T62820 CZ7A5Y 10263168 Ki > 1000000 nM T62820 CI86MW 10318576 EC50 = 380 nM T62820 CX12HM 10330132 Ki = 4800 nM T62820 CR94QY 10343566 EC50 = 878 nM T62820 CMW4B2 10353365 EC50 = 0.089 nM T62820 CZ09YG 10358265 IC50 = 20000 nM T62820 CQ1L0O 10359073 Ki = 18000 nM T62820 C6MTC4 10374869 EC50 > 1000000 nM T62820 C09LUW 10375719 IC50 > 200000 nM T62820 C29WLU 10407808 EC50 = 1823 nM T62820 C1IDG8 10413231 EC50 = 93 nM T62820 C3KHU7 10465017 EC50 > 300000 nM T62820 CK9MN4 10465478 EC50 = 40000 nM T62820 CO9MK3 10489913 EC50 > 300000 nM T62820 C34LSX 10489914 EC50 > 300000 nM T62820 C2TRI8 10492773 IC50 = 180 nM T62820 CU9BA6 10513894 EC50 > 300000 nM T62820 CQGZ24 10513895 EC50 > 300000 nM T62820 CYC9W8 10513896 EC50 > 300000 nM T62820 CG48QI 10515174 IC50 = 1100 nM T62820 CH9VN3 10560963 EC50 = 38000 nM T62820 CP0B8Q 10567792 IC50 = 240 nM T62820 C0P9JO 10587622 IC50 = 850 nM T62820 C20AXL 10607617 IC50 = 6500 nM T62820 CDN69Z 10609381 EC50 > 1000000 nM T62820 C57GCR 10656383 Ki > 1000000 nM T62820 C8FP7I 10681240 EC50 > 300000 nM T62820 C06TDU 10688450 IC50 = 220 nM T62820 CC6T7Z 10704895 EC50 > 300000 nM T62820 CC7JP9 10704896 EC50 > 300000 nM T62820 CD0E3P 10710505 IC50 = 1400 nM T62820 CBQV60 10732318 IC50 = 450 nM T62820 CC2PB0 10752213 EC50 > 300000 nM T62820 C27KWL 10752214 EC50 > 300000 nM T62820 CQTF38 10775369 EC50 = 54000 nM T62820 C6D9IL 10778385 IC50 = 1000 nM T62820 CQE5Y9 10783272 IC50 = 4360 nM T62820 C4Q3RT 10807972 IC50 = 200 nM T62820 CACY46 10826383 IC50 = 1000 nM T62820 C8MOC5 10828532 IC50 = 1800 nM T62820 C9BK1A 10846649 EC50 = 330 nM T62820 CHZ17V 10852666 IC50 = 240 nM T62820 CDO7A1 10979251 Ki = 420 nM T62820 CJ5B8P 11084869 EC50 = 7.5 nM T62820 CYP5U8 11187949 EC50 = 340 nM T62820 CSO7B4 11211597 IC50 = 25 nM T62820 CW74TN 11213605 EC50 = 186 nM T62820 CR7BZ3 11220424 EC50 = 19.8 nM T62820 C7UD6I 11235624 IC50 = 38 nM T62820 CNK6Y5 11269030 IC50 = 52 nM T62820 C7Z0HY 11271167 EC50 = 559 nM T62820 C8LSU6 11275666 EC50 = 21.2 nM T62820 CT4IL9 11281280 IC50 = 41 nM T62820 C3D0LM 11298568 Ki = 983 nM T62820 C9ASF3 11304010 IC50 = 7 nM T62820 CL1VX3 11310142 EC50 = 63.6 nM T62820 CX2T1N 11344646 EC50 = 28.6 nM T62820 C5FJ9P 11442010 IC50 = 15 nM T62820 CA50PD 11481048 Ki > 100000 nM T62820 C8N4QS 11484819 IC50 = 10 nM T62820 C8WX9P 11494153 EC50 = 4550 nM T62820 C97CIJ 11495483 EC50 = 819 nM T62820 C8P1GV 11496256 EC50 = 223 nM T62820 CYA2N5 11496550 EC50 = 442 nM T62820 C6NY5K 11503055 IC50 = 17000 nM T62820 CZF3H8 11510036 EC50 = 770 nM T62820 C9WAF1 11516962 EC50 = 782 nM T62820 CDC6P9 11530877 EC50 = 1532 nM T62820 CI3OW7 11531272 EC50 = 384 nM T62820 CTU14V 11531870 EC50 = 1500 nM T62820 CC4N0E 11537726 EC50 = 1717 nM T62820 CPA6R9 11539379 EC50 = 761 nM T62820 CQ5H1B 11543205 EC50 = 1000000 nM T62820 CB0VJ1 11545979 EC50 = 1060 nM T62820 C5JM0L 11546303 EC50 = 575 nM T62820 CW8H0Q 11559750 IC50 = 4.45 nM T62820 C3XIQ9 11559813 EC50 = 1987 nM T62820 C5TUG1 11575058 EC50 = 677 nM T62820 CHT79E 11583075 EC50 = 122 nM T62820 CGX8F6 11596869 EC50 = 201 nM T62820 CH2S1Q 11598292 EC50 = 276 nM T62820 CW3FH5 11625861 EC50 = 282 nM T62820 CZY8V2 11626305 EC50 = 676 nM T62820 CNC9T1 11626955 EC50 = 6 nM T62820 CG3YQ2 11631795 EC50 = 3273 nM T62820 CD9R3H 11633075 EC50 = 195 nM T62820 CZT84F 11646457 EC50 = 1093 nM T62820 C8YP5I 11648184 EC50 = 1160 nM T62820 C2W7YU 11648510 EC50 = 839 nM T62820 C2HBF6 11654949 EC50 = 892 nM T62820 CGKW60 11655609 EC50 = 188 nM T62820 CY59LG 11656255 EC50 = 1090 nM T62820 C3Y7PG 11656483 EC50 = 225 nM T62820 CVF97L 11663312 EC50 = 165 nM T62820 CFU63A 11663353 EC50 = 600 nM T62820 C5KEH1 11676185 EC50 = 589 nM T62820 C14GIR 11677757 EC50 = 270 nM T62820 CZ07JS 11684927 EC50 = 562 nM T62820 C8HCT2 11690041 EC50 = 5000 nM T62820 C57MBJ 11690196 EC50 = 293.5 nM T62820 CV4RD5 11691077 EC50 = 371 nM T62820 C0NU2Y 11691221 EC50 = 629 nM T62820 CBR6C9 11697718 EC50 = 291 nM T62820 CEV5N0 11699129 EC50 = 515 nM T62820 C72PVA 11710164 EC50 = 3855 nM T62820 C9ZS4H 11743092 EC50 = 3313 nM T62820 CASI54 11768848 EC50 = 10000 nM T62820 C96YUT 11820180 Ki = 23000 nM T62820 C38KRJ 11950553 EC50 = 984 nM T62820 CAQ78H 11950742 EC50 = 6367 nM T62820 C74FOC 11950744 EC50 = 1172 nM T62820 CWQ97C 11950745 EC50 = 2263 nM T62820 C4QLG1 11950746 EC50 = 3591 nM T62820 CCL2D8 11950926 EC50 = 1070 nM T62820 CB6DL5 11950927 EC50 = 559 nM T62820 CH2VY3 11951099 EC50 = 318 nM T62820 C0RP3G 11951270 EC50 = 1356 nM T62820 CY64JV 11951271 EC50 = 3544 nM T62820 CVIC83 11951272 EC50 = 1010 nM T62820 CQH10X 11951447 EC50 = 879 nM T62820 CQK7Y4 11951449 EC50 = 451 nM T62820 CAG3J7 11951806 EC50 = 228 nM T62820 CG1E3F 11951986 EC50 = 755 nM T62820 C57ARC 11951987 EC50 = 652 nM T62820 C20KVE 11951989 EC50 = 1130 nM T62820 C8NOX0 11951991 EC50 = 765 nM T62820 C84IEZ 11952168 EC50 = 598 nM T62820 CQR48X 11952169 EC50 = 779 nM T62820 CD47VA 11952347 EC50 = 788 nM T62820 CSW38G 15420544 EC50 > 10000 nM T62820 CP9Y7Q 15479143 EC50 = 0.56 nM T62820 CZ8PK5 15840277 EC50 > 1000000 nM T62820 CG3Q6X 16739372 EC50 > 1000000 nM T62820 C04GUC 17758443 Ki = 235000 nM T62820 C0Z2XO 17758444 Ki > 300000 nM T62820 CGZF13 17758445 Ki > 300000 nM T62820 C1GSZ4 17758449 Ki > 300000 nM T62820 CZW76I 17758450 Ki > 300000 nM T62820 CT64UF 17758554 Ki > 300000 nM T62820 C3X6WB 17758555 Ki > 300000 nM T62820 C1AD2J 17758556 Ki > 300000 nM T62820 CS5B7A 18138918 IC50 > 30000 nM T62820 CWEO80 18756981 Ki = 447000 nM T62820 CKX67J 18997192 EC50 > 30000 nM T62820 C5WYI2 21309795 IC50 = 312 nM T62820 CHR6P2 21393580 EC50 = 25130 nM T62820 CZ29VM 22368592 EC50 = 7810 nM T62820 C0K9DR 22884216 IC50 = 339000 nM T62820 CUB64E 23521659 EC50 = 140 nM T62820 CVMA40 23521677 EC50 = 200 nM T62820 C6X1VR 23521689 EC50 = 1100 nM T62820 CZ59GV 23521692 EC50 = 620 nM T62820 C9ZV0F 23521693 EC50 = 440 nM T62820 CRD2S7 23521697 EC50 = 36 nM T62820 CCB78W 23521698 EC50 = 180 nM T62820 CF8VY9 23521708 EC50 = 160 nM T62820 CE8Q1M 23521709 EC50 = 360 nM T62820 CK8MX3 23521713 EC50 = 1400 nM T62820 CGUN98 23521714 EC50 = 780 nM T62820 CP2SU0 23521725 EC50 = 4200 nM T62820 C8O4CW 23521727 EC50 = 1600 nM T62820 CLMX41 23521731 EC50 > 30000 nM T62820 CT9JZ3 23521734 EC50 = 2100 nM T62820 CBO38Y 23770349 EC50 = 3897 nM T62820 CDM85B 24809650 EC50 = 260 nM T62820 COM9A1 24809653 EC50 = 1170 nM T62820 C3Z2PD 24809687 EC50 = 2040 nM T62820 CSCW01 24815434 EC50 = 199.53 nM T62820 CBF6J9 24815439 EC50 = 125.89 nM T62820 C0DYP7 24815883 EC50 = 100 nM T62820 CN9AY0 24815976 EC50 = 100 nM T62820 C2A0LT 24849462 EC50 = 79.43 nM T62820 CYC98A 24849789 EC50 = 794.33 nM T62820 CB3T7C 24905650 IC50 > 1000000 nM T62820 C3BFR8 25002587 EC50 = 398 nM T62820 CB9E3V 25002939 EC50 = 390 nM T62820 CJ7KB0 25002941 EC50 = 372 nM T62820 CNK9Y0 25003298 EC50 = 347 nM T62820 CW23YC 25004010 EC50 = 174 nM T62820 CYHF64 25004352 EC50 = 186 nM T62820 CJ25HL 25008615 EC50 = 43 nM T62820 C6QGZ0 25073303 EC50 = 330 nM T62820 C9QYD4 25073615 EC50 = 1355 nM T62820 C01DRP 25173209 EC50 = 590 nM T62820 CY14JP 25173286 EC50 = 15 nM T62820 CW3PJ4 25173287 EC50 = 203 nM T62820 C43DFR 25173365 EC50 = 262 nM T62820 C4I9XA 25173448 EC50 = 117 nM T62820 CJS37O 25173616 EC50 = 7.9 nM T62820 CI0JF4 25173617 EC50 = 236 nM T62820 CRN46Z 25173691 EC50 = 75 nM T62820 CP21EC 25173697 EC50 = 84 nM T62820 C3CVG6 25173773 EC50 = 22.1 nM T62820 C7C5EF 25173776 EC50 = 142 nM T62820 CQYT89 25173778 EC50 = 76 nM T62820 CU3OL2 42610041 EC50 > 3162.28 nM T62820 C5E9CV 42610165 EC50 = 617 nM T62820 CL4R0H 42610166 EC50 = 234.42 nM T62820 CSUC90 42610167 EC50 = 2140 nM T62820 CUS06A 42629118 EC50 = 30 nM T62820 CK79XC 44155315 EC50 = 590 nM T62820 C7TXJ0 44155316 EC50 = 640 nM T62820 C65SXE 44155420 EC50 = 640 nM T62820 CQ3J6G 44155423 EC50 = 1170 nM T62820 CIU0E1 44155534 EC50 = 3820 nM T62820 CP6MG4 44155535 EC50 = 7150 nM T62820 CS6EZ9 44155538 EC50 = 640 nM T62820 CN9S0U 44155540 EC50 = 790 nM T62820 CMP31T 44155642 EC50 = 590 nM T62820 CJ49DN 44155643 EC50 = 4450 nM T62820 CK0N6G 44155644 EC50 = 1760 nM T62820 CV82HP 44155645 EC50 = 250 nM T62820 CA53BU 44155747 EC50 = 760 nM T62820 CKC0G4 44155748 EC50 = 1930 nM T62820 CQFB84 44155754 EC50 = 3300 nM T62820 C1GDO0 44155863 EC50 = 5870 nM T62820 CL94YO 44155986 EC50 = 1220 nM T62820 C5Y9DK 44155989 EC50 = 1350 nM T62820 CROL98 44156621 EC50 = 2700 nM T62820 C0TUD5 44178197 EC50 = 31 nM T62820 CNF72Q 44190035 IC50 > 10000 nM T62820 CMW71K 44285839 IC50 = 34 nM T62820 CL13FV 44302605 IC50 > 300000 nM T62820 C03QML 44302608 IC50 = 36000 nM T62820 C2H6QV 44302609 IC50 = 50000 nM T62820 CP1QS5 44302686 IC50 = 42000 nM T62820 C0V9DN 44302818 IC50 > 300000 nM T62820 CDM1P2 44302819 IC50 = 75000 nM T62820 C1GV9Q 44302837 IC50 > 300000 nM T62820 C1FJU0 44302855 IC50 > 300000 nM T62820 C34AVQ 44302856 IC50 = 37300 nM T62820 CLF56U 44302896 IC50 > 300000 nM T62820 C9Y6QA 44302913 IC50 > 300000 nM T62820 CC7BN3 44302929 IC50 > 300000 nM T62820 CKL1M8 44302930 IC50 = 61000 nM T62820 C9U0NH 44302931 IC50 = 46200 nM T62820 CD5XY2 44302932 IC50 > 300000 nM T62820 CFTA38 44322537 Ki = 1000 nM T62820 C7E8SH 44322745 Ki = 40000 nM T62820 CWV7F0 44322840 Ki = 110 nM T62820 CGL0Z3 44322843 Ki > 1000000 nM T62820 C2SKJ1 44322921 Ki = 330 nM T62820 CGK17I 44335500 EC50 = 2100 nM T62820 CB50YL 44335501 EC50 = 100 nM T62820 CZ08NT 44335514 EC50 = 1600 nM T62820 CKZ18D 44335554 EC50 = 16 nM T62820 CLK90Z 44335555 EC50 = 17 nM T62820 CZJ2H7 44335573 EC50 = 32 nM T62820 CQ1HE8 44335577 EC50 = 27 nM T62820 C7QOB9 44335578 EC50 = 18 nM T62820 CH4G8A 44335613 EC50 = 640 nM T62820 CWP53G 44335614 EC50 = 230 nM T62820 C6V3KJ 44335615 EC50 = 88 nM T62820 C4OXT1 44335626 EC50 = 29 nM T62820 CHO13Z 44335650 EC50 = 2500 nM T62820 CBY2Z8 44335670 EC50 = 310 nM T62820 C9Y6KA 44335710 EC50 > 30000 nM T62820 CHV03D 44338561 EC50 > 1000000 nM T62820 CL47OE 44345358 IC50 = 1600 nM T62820 CSZ48I 44345382 IC50 > 10000 nM T62820 CA57SX 44345536 IC50 > 10000 nM T62820 CGNR10 44345546 IC50 > 10000 nM T62820 CDRU87 44348706 IC50 = 180 nM T62820 CSJE56 44348769 IC50 = 1000 nM T62820 CUD35Q 44348846 IC50 = 190 nM T62820 C1IHR4 44348859 IC50 = 3100 nM T62820 CI06ET 44348911 IC50 = 220 nM T62820 C2O8QK 44348939 IC50 = 430 nM T62820 CM3T1Q 44348993 IC50 = 180 nM T62820 C7P2EA 44361401 Ki = 23 nM T62820 CF0LY9 44361402 Ki > 10000 nM T62820 C92YEO 44390403 EC50 = 596 nM T62820 C3ZR0Q 44392629 EC50 = 558 nM T62820 C5DUF6 44392645 EC50 = 890 nM T62820 CAS07C 44392671 EC50 = 578 nM T62820 CEZV70 44392708 EC50 = 4237 nM T62820 C90LMY 44395191 EC50 = 1418 nM T62820 CS6FD4 44395282 EC50 = 495 nM T62820 C3UGL7 44395299 EC50 = 918 nM T62820 CWZ6X4 44395327 EC50 = 241 nM T62820 C13GYT 44395381 EC50 = 7517 nM T62820 CHN13C 44397878 EC50 = 134 nM T62820 CAK39T 44406220 EC50 > 1000000 nM T62820 CH9J0V 44406221 EC50 > 1000000 nM T62820 CSD19C 44429217 EC50 > 1000000 nM T62820 CNZ16W 44429224 EC50 = 320000 nM T62820 C32RYA 44429225 EC50 > 1000000 nM T62820 CTQ29Z 44452714 IC50 = 3.49 nM T62820 CE8U7D 44452715 IC50 > 10000 nM T62820 CZG3T6 44569826 Ki > 1000000 nM T62820 CJ28TF 44569827 Ki > 1000000 nM T62820 CFZ64A 44569859 Ki > 1000000 nM T62820 CUW74T 44569860 Ki > 1000000 nM T62820 C62SAU 44591647 EC50 = 384 nM T62820 CQT61H 44591682 EC50 > 10000 nM T62820 CMP93S 44591683 EC50 > 10000 nM T62820 CA9XV2 44591684 EC50 = 5 nM T62820 CMV24G 44591685 EC50 > 10000 nM T62820 CHA08V 44591686 EC50 > 10000 nM T62820 C8FDN4 44591712 EC50 = 88 nM T62820 CC80XU 44591713 EC50 = 35 nM T62820 C80IYJ 44591714 EC50 = 280 nM T62820 CO5SY0 44591715 EC50 = 28 nM T62820 C2SEU1 44591744 EC50 = 158 nM T62820 C6F3WG 44591745 EC50 = 41 nM T62820 C2Y9IM 44591746 EC50 = 275 nM T62820 CRWM68 44591747 EC50 = 53 nM T62820 C0FY8H 44591748 EC50 = 26 nM T62820 CV5ZY0 44591770 EC50 = 97 nM T62820 CZ7ES9 44591771 EC50 = 183 nM T62820 C2OK6Y 44591772 EC50 = 32 nM T62820 CE0XV7 44591773 EC50 = 70 nM T62820 CET50O 44591774 EC50 = 4790 nM T62820 C64BTP 44591792 EC50 = 7550 nM T62820 C2ACY5 44591793 EC50 = 4380 nM T62820 CQL3J1 44591794 EC50 = 380 nM T62820 C72UIG 44591795 EC50 = 595 nM T62820 CX3T0N 44591796 EC50 = 3400 nM T62820 CJL2U9 44591797 EC50 = 1800 nM T62820 C20RKX 44591812 EC50 = 3060 nM T62820 CUJ69X 44591813 EC50 = 6360 nM T62820 CFAM64 45082292 Ki = 22387.21 nM T62820 CLBT94 46190877 EC50 = 79.43 nM T62820 CC4P3Q 46215704 EC50 = 160 nM T62820 CQ15ZS 46215708 EC50 = 501 nM T62820 CI0V4Q 46215709 EC50 = 230 nM T62820 C8ONP5 46215876 EC50 = 320 nM T62820 CCG69D 46215878 EC50 = 120 nM T62820 CNGE57 46216056 EC50 = 1660 nM T62820 C68EGY 46225320 EC50 = 316.23 nM T62820 CGH0M1 46225334 EC50 = 125.89 nM T62820 COFU37 46225335 EC50 = 199.53 nM T62820 C9XTG3 46225336 EC50 = 316.23 nM T62820 C96LBQ 46225337 EC50 = 501.19 nM T62820 C2HJY9 46225356 EC50 > 12589.25 nM T62820 CLYI35 46225357 EC50 = 63.1 nM T62820 CUTK50 46225358 EC50 = 125.89 nM T62820 C0UFE6 46225359 EC50 = 125.89 nM T62820 CS41AG 46225371 EC50 = 158.49 nM T62820 CGXJ25 46225372 EC50 = 158.49 nM T62820 CIG9F3 46225373 EC50 = 501.19 nM T62820 C4AYM0 46225374 EC50 = 794.33 nM T62820 CF1BR5 46225375 EC50 = 2511.89 nM T62820 C2REY9 46225383 EC50 = 12589.25 nM T62820 CC4Q8A 46225384 EC50 = 12589.25 nM T62820 CROL08 46225385 EC50 = 251.19 nM T62820 C9SN2I 46225386 EC50 = 50.12 nM T62820 CTI46Y 46225387 EC50 = 1995.26 nM T62820 CQK36B 46225407 EC50 = 125.89 nM T62820 CJU6S2 46225408 EC50 = 199.53 nM T62820 C6MC8Z 46225569 EC50 = 316.23 nM T62820 CS6Y9W 46225581 EC50 = 100 nM T62820 C78DON 46225582 EC50 = 158.49 nM T62820 CC8E3T 46225583 EC50 = 199.53 nM T62820 CML42B 46225584 EC50 = 39.81 nM T62820 C78MOX 46225585 EC50 > 3162.28 nM T62820 CI8C9S 46226929 EC50 = 630.96 nM T62820 CQUC74 46226930 EC50 = 977.24 nM T62820 C5F2MW 46226931 EC50 > 3162.28 nM T62820 CPEX32 46226933 EC50 > 3162.28 nM T62820 CGA3E8 46226934 EC50 = 1096.48 nM T62820 C6H1AE 46226952 EC50 = 851.14 nM T62820 CNXU31 46227786 EC50 = 158.49 nM T62820 C5KR8V 46227787 EC50 = 141.25 nM T62820 C56GKB 46227789 EC50 = 2290.87 nM T62820 CPI15K 46227790 EC50 = 645.65 nM T62820 C6K4BZ 46227792 EC50 = 446.68 nM T62820 CU9P1W 46227795 EC50 = 446.68 nM T62820 CFCB23 46227797 EC50 = 186 nM T62820 C31PAF 46700737 EC50 > 10000 nM T62820 CGS4F2 46836713 EC50 > 10000 nM T62820 CY8XU6 46887116 EC50 > 3000 nM T62820 CFZ75A 46887158 EC50 > 3000 nM T62820 CQ41EL 46887159 EC50 > 30000 nM T62820 CXRI94 46887204 EC50 > 30000 nM T62820 CD67PX 46887230 EC50 > 3000 nM T62820 C45HKB 46887231 EC50 > 3000 nM T62820 C2MF1C 46887232 EC50 > 3000 nM T62820 CWZU14 46887270 EC50 > 30000 nM T62820 CJIM29 46887271 EC50 = 1200 nM T62820 CBAG30 46887272 EC50 = 790 nM T62820 CJHM17 46887273 EC50 = 1300 nM T62820 CSO97X 46887318 EC50 > 30000 nM T62820 CQ2D0E 46887319 EC50 = 3440 nM T62820 CX8VI9 46887320 EC50 = 660 nM T62820 C8TFQ1 46887321 EC50 > 30000 nM T62820 CJ2TX5 46887322 EC50 = 360 nM T62820 CT46QN 46887367 EC50 = 590 nM T62820 CY8FH1 46887368 EC50 > 30000 nM T62820 CH9E7C 46887369 EC50 = 580 nM T62820 CQT58Z 46887370 EC50 = 360 nM T62820 CGZN85 46887371 EC50 = 350 nM T62820 CS80HA 46887372 EC50 = 240 nM T62820 CR0YT6 46887414 EC50 > 30000 nM T62820 C0H4YC 46887415 EC50 = 4110 nM T62820 CTHJ09 46887416 EC50 = 2190 nM T62820 CIBN32 46887417 EC50 = 840 nM T62820 CG03PK 46887418 EC50 = 780 nM T62820 CVIK59 46887459 EC50 > 30000 nM T62820 CF03GW 46887460 EC50 = 1180 nM T62820 CP2TE4 46887461 EC50 > 30000 nM T62820 C93HPN 46887462 EC50 > 30000 nM T62820 CT7CI1 46887463 EC50 > 30000 nM T62820 C7J3KZ 46887490 EC50 > 30000 nM T62820 CY87VO 46887491 EC50 > 30000 nM T62820 CW30ZV 46887492 EC50 > 30000 nM T62820 C4YJ6U 46887493 EC50 = 450 nM T62820 CD54VL 46887494 EC50 > 30000 nM T62820 CT50LF 46917716 EC50 = 199.53 nM T62820 CF6SM9 46917791 EC50 = 251.19 nM T62820 CJM4V9 46927956 EC50 > 50 nM T62820 CV6F9U 49799828 IC50 > 300000 nM T62820 C48MCL 49801368 Ki = 7.079 nM T62820 C5JV9D 49801369 Ki = 7.943 nM T62820 C2IS7M 49801370 Ki = 2.239 nM T62820 C49ZYG 49801371 Ki = 63.1 nM T62820 CHXD02 49822037 EC50 = 116 nM T62820 C8O0MB 49822115 Ki = 7.586 nM T62820 CET89N 49822116 EC50 = 45.7 nM T62820 C9CG2Q 49822195 EC50 = 132 nM T62820 CDC62Z 50992248 EC50 = 13 nM T62820 CN3TR7 51030965 EC50 = 159 nM T62820 CWE2O4 51033723 IC50 > 10000 nM T62820 C0L2SP 51036108 EC50 = 29 nM T62820 CAU6D5 51036701 EC50 = 430 nM T62820 CBI3A0 51036916 EC50 = 332 nM T62820 C3GQ8O 51037131 EC50 = 2200 nM T62820 CE4KP1 51050257 Ki > 10000 nM T62820 CQP6K5 51357936 EC50 = 76 nM T62820 C2DQ9V 51357937 EC50 = 3 nM T62820 C8SD6H 52941386 EC50 > 100000 nM T62820 CP97IL 52941387 EC50 > 100000 nM T62820 CN07TX 52944782 IC50 = 62000 nM T62820 CL4EM5 52947232 EC50 > 100000 nM T62820 C8JM1S 52947499 EC50 > 100000 nM T62820 CP8U6O 52948863 EC50 > 100000 nM T62820 CN1HU8 53235518 EC50 > 10000 nM T62820 CY58NO 53240406 EC50 = 5.6 nM T62820 C1WA5P 53316861 EC50 = 5011.87 nM T62820 CFGH56 53316862 EC50 = 630.96 nM T62820 CFA9L0 53317704 EC50 = 3162.28 nM T62820 COE1L6 53319016 EC50 > 10000 nM T62820 CI8V6B 53320175 EC50 = 501.19 nM T62820 CT2AE4 53320176 EC50 > 50118.72 nM T62820 CK54CE 53320818 EC50 = 398.11 nM T62820 C8XED2 53321493 EC50 = 158.49 nM T62820 CUXT69 53322147 EC50 = 1258.93 nM T62820 C30TGS 53322148 EC50 = 794.33 nM T62820 CD8L0K 53322149 EC50 = 794.33 nM T62820 CW36CH 53322382 EC50 > 10000 nM T62820 CYVT61 53323491 EC50 = 1584.89 nM T62820 CGXD80 53323492 EC50 = 630.96 nM T62820 CWQZ96 53323493 EC50 = 5011.87 nM T62820 CZJ14E 53324151 EC50 = 316.23 nM T62820 CEGK43 53324152 EC50 = 7943.28 nM T62820 CN3LP1 53324803 EC50 = 3981.07 nM T62820 CB27GO 53325450 EC50 = 630.96 nM T62820 CE45SV 53325451 EC50 = 1258.93 nM T62820 C6N0PC 53325452 EC50 = 398.11 nM T62820 CTJ85B 53325603 EC50 = 2511.89 nM T62820 C6I1SJ 53326074 EC50 = 2511.89 nM T62820 CV7Z8X 53326075 EC50 = 794.33 nM T62820 CN56WI 53326709 EC50 = 316.23 nM T62820 CCO07V 53326710 EC50 = 1995.26 nM T62820 CD2N3U 53326711 EC50 > 10000 nM T62820 CIHC67 54582001 IC50 > 30000 nM T62820 CJRG27 54761054 EC50 = 61 nM T62820 CFT41P 54761055 EC50 = 379 nM T62820 CJ8OE4 56587985 IC50 > 10000 nM T62820 CD2X1L 56651050 EC50 = 31 nM T62820 C61WQL 56968082 EC50 = 2.6 nM T62820 CYG7E8 57459475 EC50 = 696 nM T62820 CKD7Y0 57459477 EC50 = 56 nM T62820 CT70FL 57459480 EC50 = 468 nM T62820 C90COW 57459481 EC50 = 386 nM T62820 C9F4NA 57459482 EC50 = 31 nM T62820 C8Z3RY 57459483 EC50 = 299 nM T62820 C8VI3M 57459485 EC50 = 1120 nM T62820 CA2M4E 57459487 EC50 = 61.66 nM T62820 CLWD45 57459488 EC50 = 8.2 nM T62820 CC8E4J 57459494 EC50 = 6 nM T62820 CL2CK9 57459497 EC50 = 10.5 nM T62820 CEK6D7 57459500 EC50 = 116 nM T62820 CNFW08 57459501 EC50 = 24 nM T62820 CX0PZ8 57459504 EC50 = 178 nM T62820 CD2S1O 57459512 EC50 = 944 nM T62820 CH0R4N 57459517 EC50 = 149 nM T62820 CON7Q3 57459524 EC50 = 400 nM T62820 CL5DB3 57459542 EC50 = 519 nM T62820 C5S9BF 57459635 EC50 = 39 nM T62820 CH92AS 57459636 EC50 = 74 nM T62820 CH9X5W 57459640 EC50 = 102 nM T62820 C8YMH1 57459655 EC50 = 1230 nM T62820 CX0M2P 58081135 EC50 = 85 nM T62820 CBN30U 58103861 EC50 = 125 nM T62820 CKT7V5 58103890 EC50 = 150 nM T62820 CF9ID2 58966955 EC50 = 251.19 nM T62820 CCIL93 59234239 EC50 = 102 nM T62820 C4ZR5Q 59391336 EC50 = 361 nM T62820 CFCO74 59497075 EC50 = 251 nM T62820 CQ23OR 59497100 EC50 = 170 nM T62820 CW70SA 59599459 EC50 = 309.5 nM T62820 CF45DO 59599475 EC50 = 1076 nM T62820 C12XMG 59599515 EC50 = 1431 nM T62820 CIB19F 59599538 EC50 = 682 nM T62820 CC8W5L 59599545 EC50 = 87.4 nM T62820 CJIV72 59599552 EC50 = 39.3 nM T62820 C3OAM1 59599555 EC50 = 227 nM T62820 C1MJ8Z 59599565 EC50 = 470 nM T62820 CF3TQ4 59599568 EC50 = 319 nM T62820 CV91KQ 59599576 EC50 = 404.5 nM T62820 C1VAB2 59599577 EC50 = 109.6 nM T62820 CD5T6R 59599580 EC50 = 17.9 nM T62820 CHX74C 59599616 EC50 = 561.5 nM T62820 CYAQ39 60096178 EC50 = 8.37 nM T62820 C38GPO 60096183 EC50 = 26.5 nM T62820 C2NRC3 60096190 EC50 = 18.1 nM T62820 C63MKC 60096194 EC50 = 508 nM T62820 CMUL95 60096201 EC50 = 3.77 nM T62820 CW32CB 60096204 EC50 = 19.1 nM T62820 C8JAU2 60096211 EC50 = 257 nM T62820 C5PSF3 60096224 EC50 = 7.44 nM T62820 CXO4R6 60096228 EC50 = 6.32 nM T62820 C8N4UB 60096231 EC50 = 47.5 nM T62820 C9V3NZ 60096236 EC50 = 17.1 nM T62820 C38CBK 60096246 EC50 = 16 nM T62820 CN3OV8 60096250 EC50 = 6.97 nM T62820 C36ZLG 66612837 EC50 = 8510 nM T62820 CODX64 66784246 Ki = 14.79 nM T62820 C45ADN 66784262 Ki = 8.913 nM T62820 CV24AF 66784529 Ki = 3.02 nM T62820 CD7H3O 66784572 Ki = 3.631 nM T62820 CBP9O0 66784675 Ki = 11.75 nM T62820 CRFC93 66784890 Ki = 61.66 nM T62820 CQEC97 66785010 Ki = 6.761 nM T62820 C95WBM 66785027 Ki = 10.23 nM T62820 C6Q3OW 66785087 Ki = 3.631 nM T62820 CEIB16 66785101 Ki = 18.62 nM T62820 CRL4I1 66785182 Ki = 53.7 nM T62820 CBKT87 66785300 Ki = 3.89 nM T62820 CYK47D 66785393 Ki = 7.413 nM T62820 CR8QA6 66785551 Ki = 1.95 nM T62820 CDB31N 66785780 Ki = 3.162 nM T62820 C0GYH5 66786069 Ki = 5.248 nM T62820 CMD85A 66786131 Ki = 21.88 nM T62820 CB5EH8 66786493 Ki = 2.188 nM T62820 CG74XS 66786816 Ki = 6.457 nM T62820 CQE6Z9 66786902 Ki = 1.514 nM T62820 CJ1RB0 66787355 Ki = 5.012 nM T62820 COA08L 66787433 Ki = 11.75 nM T62820 CXN92C 66788653 EC50 = 55 nM T62820 C4PU9N 67056056 EC50 = 125 nM T62820 C3LDX1 67056141 EC50 = 149 nM T62820 C8YML5 67060140 EC50 = 274 nM T62820 CA2ZJ9 67060162 EC50 = 14 nM T62820 CBX67G 67246999 EC50 > 10000 nM T62820 C06MTQ 67705326 IC50 = 16.3 nM T62820 C7MLP4 67705376 IC50 = 26.1 nM T62820 CB16WU 67707808 IC50 = 18.8 nM T62820 C5K7QG 67974411 EC50 > 10000 nM T62820 CKY17T 68107697 EC50 = 1230 nM T62820 CY4OD9 68107740 EC50 = 57 nM T62820 CY49XO 68107810 EC50 = 15 nM T62820 C4SZ3V 68107813 EC50 = 9.7 nM T62820 C7VM6D 68108294 EC50 = 26 nM T62820 CA27NW 68108429 EC50 = 13.5 nM T62820 CB46KM 68108457 EC50 = 15 nM T62820 CKX84T 68108471 EC50 = 10 nM T62820 CZ7V1I 68108567 EC50 = 26 nM T62820 CFLO79 68108604 EC50 = 57 nM T62820 CZ60TR 68108857 Ki = 1.905 nM T62820 CM30YB 68109272 Ki = 38.9 nM T62820 CUQF38 68109333 Ki = 11.48 nM T62820 CZT19E 68109335 Ki = 6.026 nM T62820 CLC7E5 68109379 Ki = 61.66 nM T62820 CTYB39 68109425 Ki = 22.91 nM T62820 CH51BY 68109580 Ki = 2.042 nM T62820 CW3B2L 68109605 Ki = 10 nM T62820 CF1KB3 68109677 Ki = 6.026 nM T62820 C09TPQ 68109941 Ki = 0.8913 nM T62820 CCT07V 68290289 EC50 > 10000 nM T62820 C03JUE 68290572 EC50 > 10000 nM T62820 C8SO0Q 69092138 EC50 = 38 nM T62820 C2KV0O 69093106 EC50 = 26 nM T62820 CAQ62Y 69093344 IC50 = 7.3 nM T62820 C8IQ4U 69093439 EC50 = 37 nM T62820 CM4RD0 69093509 EC50 = 11 nM T62820 CY85RI 69093542 EC50 = 65 nM T62820 C72AHD 69093928 EC50 = 6.9 nM T62820 C0SDE4 69344751 EC50 = 251.19 nM T62820 CM1IS6 69929497 EC50 = 115 nM T62820 CZT05A 69929646 EC50 = 1286 nM T62820 CKV8E4 69929785 EC50 = 37 nM T62820 C5RI0Z 69930179 EC50 = 36 nM T62820 CG7F5Z 70051296 IC50 = 4990 nM T62820 CBK2Y6 70051926 EC50 = 1.3 nM T62820 CZ6XT7 70052526 EC50 = 7.6 nM T62820 C6PC1G 70209638 Ki = 2.57 nM T62820 C5M4GY 70681519 EC50 = 550 nM T62820 CARF46 70681520 EC50 = 1072 nM T62820 CW4MP8 70683629 EC50 = 3169 nM T62820 CEA04N 70683630 EC50 > 10000 nM T62820 CQL6G8 70683631 EC50 = 100 nM T62820 C85SZD 70685761 EC50 = 1150 nM T62820 C8ERQ5 70685762 EC50 = 363 nM T62820 C6HE1D 70685763 EC50 = 110 nM T62820 COV8Q0 70685764 EC50 = 42 nM T62820 C1X8ZL 70685765 EC50 = 832 nM T62820 CC68DO 70685766 EC50 = 275 nM T62820 CEY5P6 70685767 EC50 = 263 nM T62820 C5DM9I 70685768 EC50 = 230 nM T62820 CJSO08 70685769 EC50 = 64 nM T62820 C9KUT6 70689923 EC50 = 290 nM T62820 CGY70F 70689924 EC50 = 646 nM T62820 CRT73C 70689925 EC50 = 460 nM T62820 C3BOE9 70689926 EC50 = 1479 nM T62820 C6QGI9 70689927 EC50 = 447 nM T62820 C1I3RE 70689928 EC50 = 138 nM T62820 CLR8F3 70689929 EC50 = 100 nM T62820 CPZ9Y1 70689930 EC50 = 100 nM T62820 C9UV8C 70692086 EC50 = 479 nM T62820 CF3M0X 70694131 EC50 = 126 nM T62820 CH4JU9 70694132 EC50 = 933 nM T62820 CRP6A5 70696263 EC50 = 166 nM T62820 CB47XM 70696264 EC50 = 30 nM T62820 CXW7U0 70977933 EC50 = 148 nM T62820 CL52RS 71128783 EC50 = 531 nM T62820 CJIX85 71131322 EC50 = 0.58 nM T62820 C4JV5H 71135411 EC50 = 10.4 nM T62820 CE8L3P 71136640 EC50 = 12.4 nM T62820 CGH26Q 71136653 EC50 = 11.2 nM T62820 CW04KN 71136654 EC50 = 74 nM T62820 CAN01B 71136655 EC50 = 16.5 nM T62820 CHC91O 71137008 EC50 = 44.3 nM T62820 CH0W1O 71137010 EC50 = 13.9 nM T62820 CUB8G1 71137011 EC50 = 6.4 nM T62820 CP07IN 71137012 EC50 = 4.5 nM T62820 C28ZBK 71137034 EC50 = 11.8 nM T62820 C3N8ZO 71450118 EC50 = 501 nM T62820 CKRS61 71451227 EC50 = 330 nM T62820 CT1BS3 71454787 EC50 = 110 nM T62820 C4M0QE 71456562 EC50 = 190 nM T62820 C2R6AX 71457756 EC50 = 20 nM T62820 C0NG5K 71457757 EC50 = 4.1 nM T62820 C2D9WH 71458417 EC50 = 250 nM T62820 CV3I2G 71460259 EC50 = 710 nM T62820 C3L2SU 71461395 EC50 = 7.5 nM T62820 CKB65W 71462632 EC50 = 155 nM T62820 CNXB36 71476419 EC50 = 5.2 nM T62820 CNIW83 71479388 EC50 = 16 nM T62820 C8U0CT 71681823 EC50 = 8.2 nM T62820 CO5P1V 71681824 EC50 = 47.9 nM T62820 C6EIO9 71681825 EC50 = 12.2 nM T62820 CLH9N3 71681826 EC50 = 1170 nM T62820 CXW8R2 72714783 EC50 > 10000 nM T62820 C0HF5W 73347368 IC50 = 17000 nM T62820 CV75AO 76318478 IC50 = 132 nM T62820 CAO8Y5 76318479 IC50 = 100 nM T62820 C7L8CN 76322143 IC50 = 91 nM T62820 CG4M8N 76322144 IC50 = 89 nM T62820 C79TKZ 76332991 IC50 = 89 nM T62820 CY1V4K 76336598 IC50 = 133 nM T62820 C9J2QX 83821056 EC50 > 5000 nM T62820 CBA80Q 86691853 EC50 = 86 nM T62820 C3G4HD 86695984 IC50 = 19.9 nM T62820 CT2AF5 88593167 EC50 = 58 nM T62820 CWF97K 89497505 EC50 = 49 nM T62820 CDX7Q3 89497771 EC50 = 181 nM T62820 CFL05V 89497792 EC50 = 192 nM T62820 C3M8QU 89554892 IC50 = 146 nM T62820 C8BO4X 89735006 EC50 = 57 nM T62820 CL3AW7 89735130 EC50 = 26 nM T62820 C4RZ1G 89735186 EC50 = 70 nM T62820 C0TB9P 89735344 EC50 = 184 nM T62820 CF2UO1 89735510 EC50 = 112 nM T62820 C8FWH7 89735528 EC50 = 103 nM T62820 CC4O3J 89735530 EC50 = 80 nM T62820 C5F6VD 89735654 EC50 = 81 nM T62820 C0S7DT 89735684 EC50 = 313 nM T62820 CWZQ47 90098428 EC50 = 0.65 nM T62820 C53GQO 90668092 EC50 = 158.49 nM T62820 CZ80IY 90668093 EC50 = 125.89 nM T62820 CQ5HN3 90668094 EC50 = 251.19 nM T62820 C0X2RG 90668095 EC50 = 199.53 nM T62820 CEWD61 90668096 EC50 = 398.11 nM T62820 C0HCM5 90668097 EC50 = 158.49 nM T62820 CQ3V9Y 90668098 EC50 = 1995.26 nM T62820 C72VAL 90668099 EC50 = 316.23 nM T62820 CCG30J 90668100 EC50 = 501.19 nM T62820 CNR0U3 90668101 EC50 = 1258.93 nM T62820 C0KD7H 90668102 EC50 = 199.53 nM T62820 CLI30Z 90668103 EC50 = 251.19 nM T62820 CG1RM7 90668104 EC50 = 50118.72 nM T62820 CM2D0H 90668105 EC50 = 501.19 nM T62820 C7CN6Q 117821004 IC50 = 79.43 nM T62820 C4E9MZ 117821189 IC50 > 50118.72 nM T62820 CT7RL6 117821319 IC50 = 6.918 nM T62820 C8U9BX 117824335 IC50 = 8.913 nM T62820 C2XN3Z 117967312 EC50 = 28 nM T62820 C2CT0F 117968349 EC50 = 1.8 nM T62820 C56RJX 117968551 EC50 = 10 nM T62820 CW9RK2 117968589 EC50 = 5.5 nM T62820 CR3N4W 117971665 EC50 = 0.4 nM T62820 CA6NR3 117971683 EC50 = 13 nM T62820 C8UJ2M 117971685 EC50 = 0.5 nM T62820 C05WAR 117971699 EC50 = 6.1 nM T62820 CWN0I9 117972015 EC50 = 11 nM T62820 C9U1VQ 117972041 EC50 = 60 nM T62820 C4PY1O 117972044 EC50 = 17 nM T62820 CR6F0S 117972047 EC50 = 32 nM T62820 C3KJ0X 117972056 EC50 = 0.4 nM T62820 C7NX4A 117972153 EC50 = 16 nM T62820 C3J2TC 117972155 EC50 = 4 nM T62820 CK53MQ 117972250 Ki = 1 nM T62820 CD96PA 117972256 EC50 = 11 nM T62820 C7MP4F 118263352 EC50 = 195 nM T62820 CYZT31 118714734 EC50 = 2951 nM T62820 CVR15F 118714735 EC50 = 10715 nM T62820 CA9ZG2 118714736 EC50 = 871 nM T62820 CO69FH 118714737 EC50 = 3311 nM T62820 CW69AX 118714738 EC50 = 31623 nM T62820 C3UEW2 118714739 EC50 = 661 nM T62820 C1OCW6 118714740 EC50 = 3090 nM T62820 CR08AY 118714741 EC50 = 4677 nM T62820 C7O9PF 118714742 EC50 = 95 nM T62820 CR68DH 118714743 EC50 = 282 nM T62820 C7GXQ1 118714744 EC50 = 55 nM T62820 C6B0HF 118714745 EC50 = 178 nM T62820 CS89QO 118714746 EC50 = 355 nM T62820 CGLM54 118714747 EC50 = 81 nM T62820 C30EPW 118714748 EC50 = 141 nM T62820 COT2Z8 118714749 EC50 = 89 nM T62820 CZ4SW5 118714750 EC50 = 49 nM T62820 CGZ67Y 118714751 EC50 = 48 nM T62820 CVB84O 118714752 EC50 = 46 nM T62820 CN3Q6K 118714753 EC50 = 35 nM T62820 C4XA9K 118714754 EC50 = 98 nM T62820 CO5UN2 118714755 EC50 = 68 nM T62820 CHDR32 118714756 EC50 = 31 nM T62820 CX8W3I 118714757 EC50 = 151 nM T62820 CJ5G3Q 118718091 EC50 = 251000 nM T62820 C8SYH1 121447916 IC50 = 207 nM T62820 CUC13P 122187795 IC50 > 30000 nM T62820 CCP5U2 122195692 EC50 > 10000 nM T62820 CH2AO4 122539788 IC50 = 78 nM T62820 C1V8CY 123289788 EC50 = 1.3 nM T62820 C8RX0A 127038185 EC50 = 12870 nM T62820 CC0GA3 127038550 EC50 = 4624 nM T62820 CE0HT8 127039577 EC50 = 15 nM T62820 CS0G9A 127042771 EC50 = 191 nM T62820 CPZ70S 127052897 EC50 = 29 nM T62820 C38BRY 131801162 EC50 > 10000 nM T62820 CFC05Q 131954513 EC50 > 10000000 nM T62820 CW31CD 134129940 IC50 = 225 nM T62820 CI3PC4 134130002 EC50 = 6.8 nM T62820 C5F2YL 134130007 EC50 = 720 nM T62820 C5VEF0 134130172 EC50 = 1.7 nM T62820 C4VC9I 134130276 EC50 = 20 nM T62820 CUF61M 134130477 EC50 = 180 nM T62820 CKF21A 134130478 EC50 = 230 nM T62820 CHJF62 134130869 EC50 > 15000 nM T62820 CN74PQ 134131242 EC50 = 18 nM T62820 C0GE9K 134131273 EC50 > 3000 nM T62820 C3YM2R 134131309 EC50 = 2700 nM T62820 CNO62D 134131394 EC50 = 13 nM T62820 C28FZN 134131502 EC50 = 29 nM T62820 CL2UY8 134132133 Ki = 76 nM T62820 CP8C5N 134137754 IC50 = 34.5 nM T62820 CQT7H6 134138062 IC50 = 1130 nM T62820 CL7G4D 134139744 IC50 = 149 nM T62820 C5I6FC 134141510 IC50 = 215 nM T62820 CR4DE8 134144056 IC50 = 306 nM T62820 C5JNX4 134144441 IC50 = 280 nM T62820 CO1H6B 134152341 IC50 = 387 nM T62820 CL72ZY 134154496 IC50 = 210 nM T62820 CB8W0T 134155683 IC50 = 66.9 nM T62820 C1SFP5 134156113 EC50 = 17 nM T62820 CIR31F 134157889 EC50 = 22 nM T62820 C3EGM5 137321168 IC50 > 10000 nM T62820 CR5AB3 137634033 Ki = 595 nM T62820 C5TQS6 137635882 Ki = 1520 nM T62820 CBE4N9 137652320 Ki = 8.71 nM T62820 C48WZJ 137652500 Ki = 25.12 nM T62820 CBI4Z5 137656301 Ki = 627 nM T62820 CU2I6G 137659992 EC50 = 42.5 nM T62820 CK1ZQ3 146036859 EC50 = 10 nM T62820 C12SMP 146036860 EC50 = 140 nM T62820 CSO3M7 146036861 EC50 = 70 nM T62820 C6VB4M 146036862 EC50 = 30 nM T62820 C75DOJ 146036869 EC50 = 80 nM T62820 CHRX58 155511507 EC50 = 270 nM T62820 C7PNF3 155513095 EC50 = 50 nM T62820 CE2H9M 155514221 EC50 = 1070 nM T62820 CKYU94 155515810 EC50 = 27 nM T62820 CQN01W 155518472 EC50 = 90 nM T62820 CMTX16 155518831 EC50 = 79 nM T62820 CQ8A2I 155519573 EC50 = 190 nM T62820 C71GAL 155519836 EC50 = 141 nM T62820 CID23O 155519900 EC50 = 18 nM T62820 C5P9JY 155522079 EC50 = 600 nM T62820 CV3XK1 155523303 EC50 = 118 nM T62820 C89LOV 155524603 EC50 = 290 nM T62820 C7QRL8 155525998 EC50 = 29 nM T62820 CIE50K 155527610 EC50 = 180 nM T62820 C54IPT 155531064 EC50 = 23 nM T62820 C84PHE 155531978 EC50 = 33 nM T62820 CU87TZ 155533313 Ki = 112.2 nM T62820 CDTL70 155534303 EC50 = 15 nM T62820 C1OR2A 155535327 EC50 = 730 nM T62820 CNA3K4 155536450 EC50 = 13 nM T62820 C6BHP1 155536501 EC50 = 20 nM T62820 CYXE53 155538270 IC50 > 10000 nM T62820 CMJB23 155539343 EC50 = 210 nM T62820 CMCG93 155539952 IC50 = 45 nM T62820 CGH8T5 155540333 EC50 = 50 nM T62820 C0WE5P 155546950 EC50 = 70 nM T62820 CHK4N9 155548817 Ki = 6.166 nM T62820 CHI78O 155549028 EC50 = 71 nM T62820 CU63FZ 155550797 EC50 = 68 nM T62820 CJSF38 155551721 EC50 = 28 nM T62820 CA63SC 155552204 EC50 = 64 nM T62820 CZO03P 155552571 EC50 = 140 nM T62820 CVO21I 155553087 EC50 = 86 nM T62820 CEK92P 155554782 EC50 = 400 nM T62820 C2YX8U 155559438 EC50 = 620 nM T62820 C1GS6A 155559961 EC50 = 60 nM T62820 C3J6RS 155560108 EC50 = 2240 nM T62820 CZF2C1 155560423 EC50 = 37 nM T62820 C5G2HN 155562956 EC50 = 14 nM T62820 C5GK8N 155565811 EC50 = 70 nM T62820 CBN31S 155565817 EC50 = 18 nM T62820 C7HQ8B 155566352 EC50 = 6 nM T62820 C2KY7F 155566740 EC50 = 17 nM T62820 C6HT0Y 155567522 EC50 = 60 nM T62820 C1DML9 155567633 Ki = 4.169 nM T62820 CK4XC6 44322529 Ki = 75 nM T62820 D00EPM 73755217 IC50 > 30000 nM T62820 D00HKQ 25002940 EC50 = 316 nM T62820 D00NCL 46836562 EC50 > 10000 nM T62820 D01EAQ 11362035 EC50 = 14 nM T62820 D01EVA 6278000 Ki > 100000 nM T62820 D01YEN 1233 Ki = 110000 nM T62820 D02DEF 49765871 EC50 = 4.8 nM T62820 D03IES 44335556 EC50 = 24 nM T62820 D04DKM 104766 EC50 = 2000 nM T62820 D04GWD 59234231 Ki = 26.3 nM T62820 D04JKL 2071 Ki > 1000000 nM T62820 D04MVR 11530404 IC50 > 10000 nM T62820 D05TFE 5218788 Ki > 100000 nM T62820 D06DUE 40539 Ki = 113000 nM T62820 D06PAK 10058694 Ki = 3.9 nM T62820 D06SDD 9837317 EC50 = 0.57 nM T62820 D07GRG 10197984 EC50 = 2.69 nM T62820 D07MHL 9868580 EC50 = 27.54 nM T62820 D08BXD 9825084 EC50 = 270 nM T62820 D08CAB 83887 EC50 > 1000000 nM T62820 D08JKW 46830123 EC50 = 82 nM T62820 D08OCG 10047169 EC50 = 348 nM T62820 D09AQK 4545574 Ki > 300000 nM T62820 D09QUN 58368068 EC50 > 10000 nM T62820 D09RPR 16737207 Ki > 10000 nM T62820 D09UBS 10428048 Ki = 110 nM T62820 D09YEQ 11158623 IC50 = 14 nM T62820 D0D2GL 3972752 Ki = 11000 nM T62820 D0DX6U 23725699 IC50 > 10000 nM T62820 D0EK6P 5310984 Ki = 450 nM T62820 D0I6WA 44595851 Ki = 79.43 nM T62820 D0IO8J 3025961 Ki > 100000 nM T62820 D0J2WN 5311344 IC50 = 8000 nM T62820 D0J8OW 446355 IC50 = 4300 nM T62820 D0L0YF 4236420 EC50 > 1000000 nM T62820 D0N0NJ 15508178 IC50 = 121000 nM T62820 D0N2TP 44190040 IC50 > 10000 nM T62820 D0N9UZ 9819927 IC50 = 2.9 nM T62820 D0O1AK 23327 EC50 > 1000000 nM T62820 D0OH2P 5311040 Ki > 300000 nM T62820 D0OS8Y 15985251 IC50 > 10000 nM T62820 D0OT9B 5960 EC50 > 1000000 nM T62820 D0OV2V 6324634 IC50 = 400 nM T62820 D0P2VP 11708219 EC50 > 1000000 nM T62820 D0P3XO 5311459 Ki = 577000 nM T62820 D0PN6Z 179394 Ki = 129000 nM T62820 D0Q6VH 5311432 Ki > 100000 nM T62820 D0R0IB 56587994 IC50 > 10000 nM T62820 D0S6DK 5311455 EC50 = 48000 nM T62820 D0SL4Q 46190878 EC50 = 125.89 nM T62820 D0T5SU 158397 EC50 > 1000000 nM T62820 D0Y1WV 5310979 Ki = 110 nM T62820 D0YO8B 5311457 Ki = 84000 nM T25317 D00HPK 47641 Ki = 1500 nM T25317 D01AYJ 1549008 Ki > 50000 nM T25317 D01XBA 5035 Ki = 1 nM T25317 D06XMU 6013 Ki > 100000 nM T25317 D07BSQ 5994 Ki > 100000 nM T25317 D07KSG 2733526 Ki = 5 nM T25317 D0CT9Y 1548953 Ki = 1 nM T25317 D0D1AL 3559 Ki = 190 nM T25317 D0D7TB 9417 Ki = 13 nM T25317 D0L5WM 2157 Ki = 25 nM T25317 D0R4OM 5566 Ki = 8 nM T25317 D0Z6ST 2467 Ki = 60 nM T25317 D0I8FV 5567 Ki = 165 nM T25317 D00KVE 9907323 Ki = 1.72 nM T25317 D0K6NS 6536 Ki = 11 nM T25317 C5VS0H 10098 Ki > 100000 nM T25317 CTF7Z4 50266 Ki = 51 nM T25317 C0LQ7N 65638 Ki = 2 nM T25317 CY79XW 72027 Ki = 18 nM T25317 CN26SL 93365 Ki = 30 nM T25317 C3SG4X 185834 Ki = 1 nM T25317 CU2RH4 202478 Ki = 2200 nM T25317 CK0JI9 1548955 Ki = 2 nM T25317 C97VGU 5474589 Ki = 54 nM T25317 CFO08L 6437849 Ki = 34000 nM T25317 C2UV7A 6439331 Ki = 3 nM T25317 C1M9QS 6713949 Ki = 583 nM T25317 CD8H3W 9799239 Ki = 0.6 nM T25317 CJ96KD 9820591 Ki = 1.7 nM T25317 CXYJ93 9841596 Ki = 15 nM T25317 C78DMI 9951886 Ki = 450 nM T25317 CZ0AT6 9954083 Ki = 2 nM T25317 CQ9NP6 11198145 Ki = 5 nM T25317 CDFB43 11743300 Ki = 8500 nM T25317 CL7XE8 13998486 Ki = 39 nM T25317 CD4N5E 15163141 Ki = 1 nM T25317 C10CLM 16061352 Ki > 100000 nM T25317 CZL87E 44303090 Ki = 500 nM T25317 CX7W3K 44398003 Ki = 441 nM T25317 C2MZH9 44398036 Ki = 4 nM T25317 C7C2TW 44398114 Ki = 6 nM T25317 C17XVW 44398137 Ki = 654 nM T25317 C0N2XB 44474938 Ki = 455 nM T25317 CU63SQ 50994498 Ki = 211 nM T25317 CUL3W2 57402462 Ki = 233 nM T25317 CGKR02 71582863 IC50 = 17000 nM T25317 CZ39OQ 71583076 IC50 = 8000 nM T25317 C0RHL6 71583188 IC50 = 15000 nM T25317 CXF49Y 71583302 IC50 = 7000 nM T25317 C02KCO 71583303 IC50 = 27000 nM T25317 CYT02N 71583304 IC50 = 17000 nM T25317 CME46I 71584577 IC50 = 11000 nM T25317 CN37SA 71584578 IC50 = 7000 nM T25317 CO79PJ 73345319 Ki = 9300 nM T25317 D00FUO 4416 Ki = 0.9 nM T25317 D02WJT 7333 Ki = 6700 nM T25317 D03TNT 5753 Ki > 100000 nM T39123 D04GEI 46700761 EC50 = 5.2 nM T39123 D0P9KL 49787129 Ki = 0.036 nM T39123 CP36DZ 8478 Ki = 3600 nM T39123 C37NQO 9919540 EC50 = 3.3 nM T39123 C4SHQ7 10010442 IC50 = 16000 nM T39123 C2QEH4 10301495 Ki = 708 nM T39123 CDR52W 10328205 EC50 = 1.4 nM T39123 C7CJH5 11622248 Ki = 0.089 nM T39123 CZJ6B1 16735508 EC50 = 1.6 nM T39123 CQ6F7E 16735509 EC50 = 3.1 nM T39123 C3F1BN 16735511 EC50 = 3 nM T39123 C39KOX 16735542 EC50 = 0.99 nM T39123 CEPD53 16735543 EC50 = 1.2 nM T39123 CN80DX 16735544 EC50 = 3 nM T39123 C6JWF7 16735567 EC50 > 100 nM T39123 CQ30OG 16735729 EC50 = 1.7 nM T39123 CGR7X8 16735730 EC50 = 0.8 nM T39123 C8YW4E 16735731 EC50 = 2 nM T39123 C20VSA 16735779 EC50 = 1.3 nM T39123 CQ04DO 16735780 EC50 > 100 nM T39123 CR8GT6 16735781 EC50 = 2.7 nM T39123 CN3KA2 16736169 EC50 = 3.3 nM T39123 C4CPV9 16736170 EC50 = 1.7 nM T39123 CGS86D 16736191 EC50 = 3 nM T39123 CQJ8C7 16736192 EC50 = 2.1 nM T39123 CVQ4E2 16736193 EC50 = 1.2 nM T39123 CW3MQ4 16736392 EC50 = 4.7 nM T39123 CVZ82U 16737378 EC50 = 0.99 nM T39123 CURY37 16737730 EC50 = 5 nM T39123 C0PT2L 16738337 EC50 = 1.7 nM T39123 CM15JY 24992020 EC50 = 1.2 nM T39123 CQA87N 24993005 EC50 = 3.3 nM T39123 CJXU79 24993970 EC50 = 1.9 nM T39123 CM0VA1 24994272 EC50 = 1.8 nM T39123 C2BCY3 24994895 EC50 = 4.4 nM T39123 C43WRQ 24995205 EC50 = 2.8 nM T39123 C5FM7Y 24995518 EC50 = 1.2 nM T39123 CQ0AX6 24995519 EC50 = 5.2 nM T39123 C10SWN 24996155 EC50 = 2.3 nM T39123 CMG2H1 24996486 EC50 = 1.6 nM T39123 CT6PL0 24996487 EC50 = 4.9 nM T39123 C70UHN 24996490 EC50 = 0.43 nM T39123 CL1UD5 24996809 EC50 = 1.1 nM T39123 CK17PD 24996810 EC50 = 2.4 nM T39123 C52IBC 25075960 EC50 = 0.56 nM T39123 CL34UW 25075963 EC50 = 0.65 nM T39123 CIO6F0 25075965 EC50 = 1.4 nM T39123 COI6C1 25075973 EC50 = 0.47 nM T39123 CA89SK 25075978 EC50 = 5.2 nM T39123 CH9NM7 25084920 EC50 = 0.073 nM T39123 C36SXI 25084922 EC50 = 2.8 nM T39123 C6S2CB 25138123 IC50 = 0.12 nM T39123 C0APO3 25138124 EC50 = 2.5 nM T39123 C8RYH9 25138125 EC50 = 5.4 nM T39123 CV8O2Q 25138126 IC50 = 32 nM T39123 CPF6T8 25138127 IC50 = 460 nM T39123 CZL08E 25138128 IC50 = 380 nM T39123 CLE2X9 25138129 EC50 = 4.3 nM T39123 CAG05L 25138130 IC50 = 32 nM T39123 CRBW20 25138131 IC50 = 0.24 nM T39123 C0XMG1 25138132 IC50 = 240 nM T39123 CA58FK 44419644 Ki = 82.7 nM T39123 C5LYA4 44419664 Ki = 10000 nM T39123 CEM4B9 44419672 Ki = 9.4 nM T39123 CK9I3C 44419676 Ki = 88.1 nM T39123 C5SU4A 44419677 Ki = 10000 nM T39123 C3NX6G 44425065 EC50 = 3.1 nM T39123 CETO79 46906646 IC50 > 30000 nM T39123 CXWN52 46906647 IC50 = 890 nM T39123 CY4L2G 53318788 IC50 > 30000 nM T39123 CSGI29 57653049 EC50 = 0.75 nM T39123 C32WXO 57653056 EC50 = 2.3 nM T39123 CQ3E0F 71449398 EC50 = 0.24 nM T39123 CVNR92 71449399 Ki = 0.12 nM T39123 CRM3V8 71449427 EC50 = 0.023 nM T39123 C5HTR3 71449428 EC50 = 0.36 nM T39123 C4ZNW1 71449429 EC50 = 0.15 nM T39123 CM5F3O 71451197 EC50 = 0.11 nM T39123 CG85XR 71451222 EC50 = 1.5 nM T39123 CSL41G 71451223 EC50 = 0.33 nM T39123 CSJ9V7 71453041 EC50 = 0.13 nM T39123 CF6TH4 71454755 EC50 = 0.041 nM T39123 CDE4V6 71454783 EC50 = 0.065 nM T39123 CTKG87 71454784 EC50 = 3.9 nM T39123 C8MU2C 71456524 IC50 = 0.61 nM T39123 CDQ5R8 71456525 IC50 = 0.49 nM T39123 C4PGM7 71456556 EC50 = 1.4 nM T39123 CH08JC 71456557 EC50 = 0.32 nM T39123 C2O4EW 71458409 EC50 = 7.2 nM T39123 CJN7H4 71458410 EC50 = 0.27 nM T39123 C6OFU9 71458411 EC50 = 76 nM T39123 C15TJE 71458412 EC50 = 0.29 nM T39123 C53GHV 71460218 EC50 = 0.13 nM T39123 C6UF1I 71460219 EC50 = 0.1 nM T39123 CCD8U3 71460220 EC50 = 0.098 nM T39123 CKUG49 71460251 EC50 = 5.8 nM T39123 C59CNG 71460252 EC50 = 0.029 nM T39123 C7AXG0 71460253 EC50 = 0.34 nM T39123 C8B3OF 71460254 EC50 = 1.4 nM T39123 C8FA9K 71461936 Ki = 0.046 nM T39123 C0IL1S 71461937 IC50 = 0.51 nM T39123 CC8AD0 71461938 EC50 = 0.05 nM T39123 CV7N6I 71461939 EC50 = 0.24 nM T39123 CJV5K8 71461940 EC50 = 0.072 nM T39123 CFX17J 71461962 EC50 = 0.039 nM T39123 C1XEW4 71461963 EC50 = 10 nM T39123 CRPE69 72711369 Ki = 0.045 nM T39123 C9DYJ7 72711370 Ki = 0.062 nM T39123 C19QVF 72711589 Ki = 0.086 nM T39123 C5UPE8 72711802 Ki = 0.12 nM T39123 CYT42N 72711803 Ki = 0.055 nM T39123 C2JD9A 72712017 Ki = 0.29 nM T39123 CN16AD 72712018 Ki = 0.11 nM T39123 CCJ3Q2 72712230 Ki = 0.052 nM T39123 CRJF51 72712231 Ki = 0.51 nM T39123 CV60KA 72712449 Ki = 0.12 nM T39123 CO1E6F 72712450 Ki = 0.2 nM T39123 C47VKG 72712666 Ki = 0.21 nM T39123 C95OKS 72712667 Ki = 0.044 nM T39123 C2E3SM 72712870 Ki = 0.21 nM T39123 COGF32 72712871 Ki = 0.2 nM T39123 CT4H1A 72713068 Ki = 0.12 nM T39123 CBNS46 72713069 Ki = 0.086 nM T39123 CY40CT 72713283 Ki = 0.032 nM T39123 C74TQW 72713284 Ki = 0.065 nM T39123 CG56KH 72713503 Ki = 0.2 nM T39123 CG1Z9Y 72713504 Ki = 0.11 nM T39123 C4VM7N 90324505 EC50 = 0.07 nM T39123 C3S1VA 90324512 EC50 = 120 nM T39123 C2AY1B 90324535 EC50 = 0.07 nM T39123 C6OKG1 90488921 EC50 = 2.5 nM T39123 C8EBD0 118707476 Ki = 0.074 nM T39123 CZ9FT5 118707477 Ki = 0.086 nM T39123 C6AUZ9 118707478 Ki = 0.052 nM T39123 C57NZB 118707479 EC50 = 4.4 nM T39123 CFD65J 118707480 EC50 = 1.5 nM T39123 CN1LZ9 118707481 EC50 = 0.59 nM T39123 C18IBL 118707482 Ki = 0.096 nM T39123 CGVP49 118707483 EC50 = 2.8 nM T39123 CJ4N0R 118707484 Ki = 0.037 nM T39123 CO3MI9 118707485 Ki = 0.036 nM T39123 C1WIM0 118707486 Ki = 0.028 nM T39123 CYV39R 118707487 Ki = 0.2 nM T39123 CPOR71 118707488 EC50 = 1.3 nM T39123 C35SAG 118707489 EC50 = 0.49 nM T39123 CO46GB 118707490 EC50 = 0.63 nM T39123 CJ24EG 118707491 Ki = 0.12 nM T39123 CR7O5H 118707492 Ki = 0.039 nM T39123 CF42GO 118707493 EC50 = 0.8 nM T39123 C91JFU 118707494 Ki = 0.034 nM T39123 CRVI37 118707495 Ki = 0.027 nM T39123 C9T0QG 118707496 Ki = 0.089 nM T39123 CT8S3P 118707497 Ki = 0.038 nM T39123 CD0WC6 118708107 Ki = 0.026 nM T39123 C7TXJ1 118735592 EC50 = 0.6 nM T39123 CV67KT 118735593 EC50 = 0.006 nM T39123 C7GMR6 118735594 EC50 = 0.9 nM T39123 C6B9SG 118735595 EC50 = 0.1 nM T39123 CHW34M 118735596 EC50 = 0.08 nM T39123 C5X7QV 118735679 EC50 = 13.9 nM T39123 C68ZHV 118735680 EC50 = 7.2 nM T39123 C1G0AZ 118735681 EC50 = 182 nM T39123 CFJ68R 118735682 EC50 > 500 nM T39123 CW5Y1F 118735683 EC50 = 2.9 nM T39123 C12CFY 118735684 EC50 = 24.4 nM T39123 CE1LW7 118735685 EC50 = 1.6 nM T39123 CU61JE 118735686 EC50 = 216 nM T39123 C4EDS9 134132372 EC50 = 0.48 nM T39123 CLCJ20 134135834 EC50 = 2.7 nM T39123 CP24SX 134143614 EC50 = 3.6 nM T39123 CP5FD6 134150351 EC50 = 0.49 nM T39123 C2WXP1 134150893 EC50 = 5.8 nM T39123 CV3ZI2 134151953 EC50 = 2 nM T39123 CW95DP 134154824 EC50 = 1.9 nM T39123 CI3OY0 134157013 EC50 = 0.61 nM T39123 CU37XC 134157281 EC50 = 22 nM T39123 C30FKQ 134157735 EC50 = 5.5 nM T39123 CH7OX8 135401501 IC50 = 3.6 nM T39123 CJ6N0V 135410889 IC50 = 10 nM T39123 CGEL62 135410891 IC50 = 25 nM T39123 C8U0TV 135528869 IC50 = 2100 nM T39123 CF0Z2T 135936864 IC50 = 1100 nM T39123 CR71AU 135936875 IC50 = 3.7 nM T39123 COQU30 136016359 IC50 = 24000 nM T39123 CR5X2P 136016360 IC50 = 34 nM T39123 CJR7Q3 136016361 IC50 = 33000 nM T39123 C1Z7SR 136016362 IC50 = 30 nM T39123 CG1HK6 136016372 IC50 = 120 nM T39123 C0PDO9 136016373 IC50 = 490 nM T39123 CQ47XG 136016379 IC50 = 480 nM T39123 CZVA18 136016380 IC50 = 7.4 nM T39123 CT73EU 136016381 IC50 = 9.8 nM T39123 CW5C9G 136016382 IC50 = 19 nM T39123 C7N9GK 136016389 IC50 = 12 nM T39123 C1QX4H 136016390 IC50 = 120 nM T39123 CKE02M 136016391 IC50 = 14 nM T39123 CMO0T8 136016392 IC50 = 45 nM T39123 C2HO5R 136016397 IC50 = 31 nM T39123 C97USJ 136016398 IC50 = 15 nM T39123 CF4B8O 136016399 IC50 = 32 nM T39123 CK8RP5 136016406 IC50 = 32 nM T39123 CTF9P2 136016407 IC50 = 8 nM T39123 CWI8P3 136016412 IC50 = 11 nM T39123 CKGQ75 136016413 IC50 = 1200 nM T39123 C0AQ7F 136016436 IC50 = 1500 nM T39123 C6X2DT 136016437 IC50 = 9900 nM T39123 C27HJQ 136016443 IC50 = 570 nM T39123 C1SLG4 136016444 IC50 = 51 nM T39123 CIAW82 136016471 IC50 = 180 nM T39123 C4X6FN 136016472 IC50 = 4.6 nM T39123 C2A3NT 136016473 IC50 = 10 nM T39123 CB62WX 136016474 IC50 = 10 nM T39123 CZ1M4G 136016475 IC50 = 16 nM T39123 C30HUY 136016476 IC50 = 10 nM T39123 C3E0AK 136016477 IC50 = 18 nM T39123 CBN5P4 136016478 IC50 = 17 nM T39123 C65OCQ 136016479 IC50 = 8 nM T39123 CJNO30 136016480 IC50 = 22 nM T39123 CT3M4D 136016481 IC50 = 9.7 nM T39123 C60IKA 136016482 IC50 = 7.9 nM T39123 C5T4QK 136016483 IC50 = 18 nM T39123 CIF8U7 136016484 IC50 = 14 nM T39123 CAFQ17 136016486 IC50 = 20 nM T39123 CYB5V3 136016487 IC50 = 4.1 nM T39123 CP67NX 136016488 IC50 = 8.4 nM T39123 C6S5WT 136016489 IC50 = 16 nM T39123 CGLB52 136016490 IC50 = 12 nM T39123 C80OZB 136016491 IC50 = 30 nM T39123 C6FPZ0 136016492 IC50 = 15 nM T39123 CL8G2K 136016493 IC50 = 30 nM T39123 CSIC76 136016517 IC50 = 7.3 nM T39123 CX94OU 136016518 IC50 = 15 nM T39123 C7I4EX 136016519 IC50 = 11 nM T39123 C9DES8 136016521 IC50 = 9.7 nM T39123 C6VIE8 136016522 IC50 = 18 nM T39123 CXM7G2 136016523 IC50 = 20 nM T39123 CJEY60 155514052 EC50 = 0.17 nM T39123 CS0K9I 155518633 EC50 = 0.89 nM T39123 C5MIX2 155522287 EC50 = 0.058 nM T39123 CFH80A 155527587 EC50 = 0.13 nM T39123 CKL19Y 155529496 EC50 = 0.62 nM T39123 C0WQA2 155529648 EC50 = 0.028 nM T39123 C9TNM5 155533419 EC50 = 0.27 nM T39123 C3DY9F 155534572 EC50 = 7.7 nM T39123 CXH7J8 155534639 EC50 = 0.23 nM T39123 C7W0RS 155535993 EC50 = 1.4 nM T39123 C05WMX 155536247 EC50 = 0.11 nM T39123 C1Z6WR 155538456 EC50 = 0.6 nM T39123 C3H6MD 155541282 EC50 = 1.5 nM T39123 C2M6UZ 155545453 EC50 = 0.037 nM T39123 C0F5ZQ 155547611 EC50 = 130 nM T39123 CQ6OT8 155547823 EC50 = 0.024 nM T39123 C1F2AE 155548337 EC50 = 0.16 nM T39123 CZ21YV 155549139 EC50 = 0.24 nM T39123 CO8GB1 155550061 EC50 = 0.022 nM T39123 C1J4YQ 155550676 EC50 = 2.1 nM T39123 C7PS9D 155551159 EC50 = 0.068 nM T39123 C3ZJ1N 155554573 EC50 = 0.33 nM T39123 CRQ10Z 155559289 EC50 = 0.13 nM T39123 CA1R6T 155559308 EC50 = 8.2 nM T39123 C06LPU 155565826 EC50 = 0.12 nM T39123 CW5M4U 16735568 EC50 = 1 nM T39123 D01VSI 25240297 Ki = 0.035 nM T39123 D08UWO 53320361 IC50 = 830 nM T39123 D0JE3Z 16735569 EC50 = 0.45 nM T84791 C5Z1QA 96028 IC50 = 10300 nM T84791 C0ZI3J 11298263 IC50 > 100000 nM T84791 CKI97Z 12344252 IC50 = 25100 nM T84791 CKSL53 12507616 IC50 = 2900 nM T84791 COF8W3 13008156 IC50 = 1600 nM T84791 CGW49I 25146686 IC50 = 7100 nM T84791 C84YXH 74763382 IC50 > 30000 nM T84791 C7S6YM 90348686 IC50 = 11000 nM T84791 CAZ6F3 123132902 IC50 = 60 nM T84791 CP60WQ 126599605 IC50 = 15000 nM T84791 CL9DA5 126599606 IC50 = 30000 nM T84791 CIM95P 126599607 IC50 > 100000 nM T84791 CZM3T2 126599609 IC50 = 7000 nM T84791 CBZ9G6 126599610 IC50 > 100000 nM T84791 CD57UE 126599615 IC50 > 100000 nM T84791 C05JCQ 126599616 IC50 > 50000 nM T84791 C27LVH 126599619 IC50 = 24000 nM T84791 CQ4OX7 126599621 IC50 = 6900 nM T84791 CU9IB6 126599623 IC50 = 15300 nM T84791 C50GVU 126599624 IC50 < 500 nM T84791 CE4U8C 126599625 IC50 = 4000 nM T84791 C3NUF1 126599626 IC50 = 7000 nM T84791 CG5JH7 126599627 IC50 = 500 nM T84791 CH8TE6 126599628 IC50 = 20000 nM T84791 CAY4G6 126599629 IC50 = 41000 nM T84791 CEQ96X 126599630 IC50 = 68000 nM T84791 CY86ZU 126599632 IC50 = 16000 nM T84791 CF35OY 126599634 IC50 = 18000 nM T84791 C0X4TK 126609831 IC50 > 100000 nM T84791 CQ9KN4 129892190 IC50 = 5.8 nM T84791 C43MXV 137644429 IC50 = 300 nM T84791 CRD19U 137644814 IC50 > 100000 nM T84791 C97ABQ 137644943 IC50 > 100000 nM T84791 C97MXP 137648465 IC50 > 100000 nM T84791 C2JPC1 137656599 IC50 = 35000 nM T09395 CBZ7P2 2928097 Ki = 49 nM T09395 CERF41 3151315 Ki = 1120 nM T09395 CL4GK5 13686033 IC50 = 6755 nM T09395 CY5SQ3 13755302 IC50 = 0.01 ug.mL-1 T09395 C2WEO7 44332503 IC50 = 0.05 ug.mL-1 T09395 C1XHA3 44332504 IC50 = 0.04 ug.mL-1 T09395 CN2K5O 44332505 IC50 = 0.01 ug.mL-1 T09395 CC47JX 44332506 IC50 = 0.04 ug.mL-1 T09395 CX83UG 118165178 IC50 > 100000 nM T09395 CWX3Z7 118165190 IC50 > 100000 nM T09395 C3S5OA 118165200 IC50 = 105 nM T09395 C95RGM 118165205 IC50 = 23100 nM T09395 C3Y0TE 118165222 IC50 > 100000 nM T09395 CE9Z3K 118165243 IC50 = 163 nM T09395 C2VZW7 118165257 IC50 = 385 nM T09395 CIJN30 118165260 IC50 = 765 nM T09395 CA8YG6 118165270 IC50 > 100000 nM T09395 C84VSY 118165287 IC50 = 123 nM T09395 C6X5HK 118165290 IC50 = 36 nM T09395 CNFT52 118165293 IC50 > 100000 nM T09395 CB59GF 118165313 IC50 = 175 nM T09395 CFIV09 118165354 IC50 = 389 nM T09395 CZ8RQ9 118165413 IC50 = 1011 nM T09395 C3F6XG 118165440 IC50 = 232 nM T09395 CWI08V 118165445 IC50 = 4160 nM T09395 CA9E0U 118165472 IC50 = 1525 nM T09395 CDAC50 118165497 IC50 = 384 nM T09395 CWP90I 118165555 IC50 > 100000 nM T09395 CM6JI8 118165621 IC50 = 945 nM T09395 C8V1IU 118165625 IC50 = 1175 nM T09395 CNPW85 118165709 IC50 = 149 nM T09395 CAZ25P 118165748 IC50 = 2255 nM T09395 C65DLT 118165752 IC50 > 100000 nM T09395 CA9UQ1 118165756 IC50 = 123 nM T09395 CATZ25 118165760 IC50 > 100000 nM T09395 CN4O5K 118165763 IC50 = 84 nM T09395 CR5HV8 121410292 IC50 = 870 nM T09395 CVE96K 121410294 IC50 = 495 nM T09395 CK9G7V 121410328 IC50 = 1800 nM T09395 CQ3KL4 121410329 IC50 = 1430 nM T09395 CBN62U 121410340 IC50 = 1900 nM T09395 CNF06J 121410352 IC50 = 1200 nM T09395 CR70JL 126641909 IC50 = 41 nM T09395 CT7M6Q 126641926 IC50 = 82 nM T09395 CLG67Z 126641948 IC50 = 48 nM T09395 CVAC39 126641974 IC50 = 580 nM T09395 C1ZTB7 126641995 IC50 = 44 nM T09395 CA81IH 126642266 IC50 = 47 nM T09395 CNJL38 126642277 IC50 = 59 nM T09395 CIW02N 126642282 IC50 = 87 nM T09395 CO09EN 155514507 IC50 = 180 nM T09395 CGWL21 155515495 IC50 = 1850 nM T09395 CPZ1J2 155515757 IC50 = 530 nM T09395 CVS35D 155518925 IC50 = 395 nM T09395 CS0ER5 155528109 IC50 = 330 nM T09395 C2WPD6 155530588 IC50 = 21 nM T09395 CYH2Z6 155530878 IC50 = 145 nM T09395 CGKM58 155542422 IC50 = 44 nM T09395 CN9LP5 155551221 IC50 = 27 nM T09395 CGV1M3 155552611 IC50 = 505 nM T09395 CM5VI1 155561970 IC50 = 19500 nM T94879 D05MQK 110635 IC50 = 1.2 nM T94879 D0C9SY 135400189 Ki = 0.7 nM T94879 D0F9GE 3108 IC50 = 574 nM T94879 D0NJ3V 4680 IC50 = 8800 nM T94879 D0Y5JC 9869929 Ki = 5 nM T94879 D0Y9ZE 4197 IC50 = 740 nM T94879 D0Z7ZM 135398744 Ki = 1.6 nM T94879 D03QJL 3671 IC50 = 103000 nM T94879 D05OQG 5318997 IC50 = 5900 nM T94879 D09OCK 135430955 IC50 = 4.2 nM T94879 D0A9IY 135564558 IC50 > 10000 nM T94879 D0L0BX 5318980 IC50 = 2200 nM T94879 D0M9FQ 11465695 IC50 = 0.5012 nM T94879 D0T5PO 5092 IC50 = 720 nM T94879 D05VBJ 71295299 IC50 > 10000 nM T94879 D0WS3T 72706254 IC50 = 260 nM T94879 D00SPK 23665864 IC50 = 3.7 nM T94879 D00YPW 135399235 Ki = 130 nM T94879 D01QUF 9842576 Ki > 100000 nM T94879 D02EMR 151170 IC50 > 10000 nM T94879 D05VLN 55690 IC50 = 58000 nM T94879 D0BK6B 3021729 IC50 > 10000 nM T94879 D0F0CS 5723 IC50 > 10000 nM T94879 D0K2BQ 71356 Ki = 7500 nM T94879 D0N5SC 135536943 IC50 = 1.23 nM T94879 D0W8OH 135529458 IC50 = 80 nM T94879 CVQ0G5 1348 IC50 = 500 nM T94879 C03NGJ 1713 IC50 = 230 nM T94879 CH8J2B 4977 Ki = 600000 nM T94879 CCJ8F0 5353 IC50 = 21000 nM T94879 C3B8VG 5369 IC50 = 1 nM T94879 CAMB41 100554 IC50 = 5500 nM T94879 C9T3FB 105007 IC50 = 1580 nM T94879 CGA17S 127779 Ki = 6500 nM T94879 C1H8NR 155248 IC50 > 50000 nM T94879 CH2P8A 158961 Ki = 600000 nM T94879 CVN23X 158962 Ki = 600000 nM T94879 CL27HC 160179 IC50 = 9300 nM T94879 CYWS98 185848 IC50 > 40000 nM T94879 C78DLE 205964 IC50 = 360 nM T94879 C1B6ZL 662965 IC50 > 50000 nM T94879 C3A4HW 675226 IC50 = 8600 nM T94879 CA56MW 675227 IC50 = 3900 nM T94879 CHAB75 696516 IC50 = 1900 nM T94879 CW2U6N 698956 IC50 = 420 nM T94879 CYBA13 719250 IC50 = 4700 nM T94879 C1HM0K 832282 IC50 = 4300 nM T94879 C9KVI7 832283 IC50 = 22000 nM T94879 CM6Q1D 869895 IC50 = 2400 nM T94879 C6QBR5 874599 IC50 = 540 nM T94879 CR7A3U 930420 IC50 = 1200 nM T94879 CWIA36 987187 IC50 = 5600 nM T94879 CT62PH 987189 IC50 = 3100 nM T94879 CO0Z8N 1002275 IC50 = 1700 nM T94879 CXQ4P8 1183964 IC50 = 860 nM T94879 CZQ09F 1204882 IC50 = 7200 nM T94879 CHP0S3 1204883 IC50 = 570 nM T94879 C0JM2Q 1215407 IC50 = 700 nM T94879 CZ2XI5 1271431 IC50 = 3100 nM T94879 COW58U 1277329 IC50 = 190 nM T94879 C6VF0S 1490272 IC50 = 840 nM T94879 CQ69OY 1490552 IC50 = 1100 nM T94879 CD0G9E 1553819 IC50 = 14000 nM T94879 CYD6E3 1553838 IC50 = 190 nM T94879 CXP17G 1604254 IC50 = 4600 nM T94879 C8JLO0 2243267 IC50 = 370 nM T94879 CTQ23N 2452792 IC50 = 800 nM T94879 CLNU08 2456309 IC50 = 740 nM T94879 CYP23V 2465033 IC50 = 800 nM T94879 CE70KT 2471983 IC50 = 1200 nM T94879 CE4D1W 2789492 IC50 = 5600 nM T94879 CFC30O 2789499 IC50 = 1000 nM T94879 C4LSR7 2886111 IC50 > 10000 nM T94879 C6AT3L 2930929 IC50 = 6300 nM T94879 CD70ZG 3119958 IC50 = 8700 nM T94879 C4MSC9 3120507 IC50 = 3000 nM T94879 CPX4V3 4352680 IC50 = 130620 nM T94879 C5IZS9 4636426 IC50 = 746450 nM T94879 CC3LA4 4672917 IC50 = 8500 nM T94879 C5P0LU 4672918 IC50 = 29300 nM T94879 C3JHM8 4687521 IC50 = 1.2 nM T94879 C0JVX6 4867627 IC50 = 4900 nM T94879 CN0Z3D 4880961 IC50 = 11000 nM T94879 C0C9HP 6610310 IC50 = 19 nM T94879 CAYS61 6918354 IC50 = 4000 nM T94879 CB40PM 6918356 IC50 = 200 nM T94879 CI7K0P 6918667 IC50 = 69800 nM T94879 CP1GO7 6918668 IC50 > 84900 nM T94879 CA05PF 6918674 IC50 = 700 nM T94879 C87WYR 6918795 IC50 > 67300 nM T94879 CRGE51 6918796 IC50 > 101000 nM T94879 CUP4M8 6918797 IC50 > 50700 nM T94879 C0LRO8 6918798 IC50 > 101000 nM T94879 C53ESK 6918799 IC50 > 91000 nM T94879 CU1E0G 6918800 IC50 > 101000 nM T94879 CRU46D 7161211 IC50 = 3250 nM T94879 CQ41MA 8055545 IC50 = 2300 nM T94879 CZF0N3 8055573 IC50 = 2400 nM T94879 CN86QP 8078832 IC50 = 2500 nM T94879 CI15SH 9797222 IC50 = 14000 nM T94879 CNC2F4 9798336 IC50 > 1000000 nM T94879 CFJ62Y 9799389 IC50 > 10000 nM T94879 CZH08Y 9802738 IC50 = 7.2 nM T94879 CDV76T 9803328 Ki = 0.29 nM T94879 CR09LM 9805655 IC50 = 0.3 nM T94879 CB57DJ 9807085 IC50 = 72 nM T94879 CXF0J7 9818343 IC50 = 10 nM T94879 C1CXA5 9818702 IC50 = 5000 nM T94879 CSOX21 9819114 IC50 = 2.8 nM T94879 C1MN3A 9821924 IC50 = 2 nM T94879 C7FY1U 9824408 IC50 = 1.1 nM T94879 C4J2XE 9836643 IC50 > 101000 nM T94879 C4YB1S 9844037 IC50 = 5.3 nM T94879 C5YQB0 9859898 IC50 = 78000 nM T94879 CZGM43 9864862 IC50 = 22000 nM T94879 CEI5P4 9868140 IC50 = 440 nM T94879 C92GMV 9879320 IC50 = 13000 nM T94879 C0Q5VN 9880010 IC50 > 101000 nM T94879 CWD1F6 9880288 IC50 > 101000 nM T94879 C2NK8E 9888568 IC50 = 0.56 nM T94879 C0P8ZH 9892886 Ki = 0.21 nM T94879 CC05QE 9901606 IC50 = 101000 nM T94879 CMBO89 9912467 IC50 = 2000 nM T94879 CBA29H 9922545 IC50 > 101000 nM T94879 CKF4C2 9922691 IC50 = 73200 nM T94879 CY17NM 9922999 IC50 = 8400 nM T94879 C70AMC 9924305 IC50 = 7270 nM T94879 CKI6N2 9924468 IC50 > 88000 nM T94879 C6AZ5F 9924709 IC50 > 101000 nM T94879 C54ICU 9927654 IC50 = 3500 nM T94879 C60BWM 9933503 IC50 = 0.8 nM T94879 CX1UV7 9946954 IC50 = 20160 nM T94879 C7OP5A 9947052 IC50 = 3970 nM T94879 C04HAV 9949594 IC50 = 225 nM T94879 C53AVJ 9951793 IC50 = 2.3 nM T94879 CE8ZD7 9954790 IC50 = 0.93 nM T94879 CH46TF 9954942 Ki = 0.23 nM T94879 C8X7RN 9956576 IC50 = 0.1 nM T94879 C2OYA1 9957043 IC50 = 0.55 nM T94879 CJO0X4 9966737 IC50 = 10940 nM T94879 CFP1Y5 9966830 IC50 > 101000 nM T94879 C9NKY4 9967652 IC50 = 74000 nM T94879 CI6AX1 9968005 IC50 > 101000 nM T94879 C7PCS8 9968050 IC50 = 40350 nM T94879 CFB48Q 9968370 IC50 = 98000 nM T94879 CU73AJ 9968471 IC50 > 101000 nM T94879 C0AP8O 9969020 IC50 = 17880 nM T94879 C9X7PF 9972372 IC50 = 8800 nM T94879 CL6V2I 9973407 IC50 = 770 nM T94879 CCDX84 9973586 IC50 = 0.53 nM T94879 C5AE2I 9973597 IC50 > 200000 nM T94879 CTQ59Y 9975543 IC50 = 3600 nM T94879 CW3S7O 9977675 IC50 > 1000000 nM T94879 C05RPA 9977814 IC50 = 2700 nM T94879 C20XIY 9985391 IC50 = 2200 nM T94879 CHG4K5 9992525 IC50 = 64000 nM T94879 CO87TV 9994528 IC50 = 100 nM T94879 CC86WM 9995163 IC50 = 6800 nM T94879 CB9EY5 9995187 IC50 = 90 nM T94879 CWJ0K5 9995367 IC50 = 210 nM T94879 CZR07N 9995467 IC50 = 930 nM T94879 C3GHJ7 9996490 IC50 = 105 nM T94879 CH70VI 9996675 IC50 = 1100 nM T94879 CE5O4D 9998316 IC50 = 350 nM T94879 CYS20P 10004422 IC50 = 38000 nM T94879 CB41WF 10017397 IC50 = 3000 nM T94879 CKE92N 10017795 IC50 = 3600 nM T94879 CHJ73C 10018556 IC50 = 8700 nM T94879 CI9WK7 10021158 IC50 = 1300 nM T94879 C6MUC5 10024867 IC50 = 2500 nM T94879 C5E4QJ 10030897 Ki = 0.24 nM T94879 C1G5XC 10032458 IC50 = 6500 nM T94879 CE25WO 10039122 IC50 = 4400 nM T94879 CUYW65 10039809 IC50 = 20000 nM T94879 C0SZB8 10039848 IC50 = 36300 nM T94879 CJ1Q7Z 10040540 IC50 = 50 nM T94879 CJ05CZ 10040882 IC50 = 15000 nM T94879 CK5VB0 10041530 IC50 = 14000 nM T94879 C9FD1X 10041853 IC50 = 7500 nM T94879 CT6Y9J 10043209 IC50 > 1000000 nM T94879 CY6FQ4 10053217 IC50 = 3 nM T94879 CD1N4K 10062262 IC50 = 1000 nM T94879 CHCJ86 10065791 IC50 = 810 nM T94879 CC6PO8 10066654 IC50 > 40000 nM T94879 C3MA2L 10067044 IC50 > 1000000 nM T94879 C5FCT6 10070215 IC50 = 0.6 nM T94879 COSV65 10074226 Ki = 0.23 nM T94879 CG39NX 10083598 IC50 = 40000 nM T94879 C5P7AS 10083609 IC50 = 6000 nM T94879 C7YBR0 10083610 IC50 = 33000 nM T94879 CAX67L 10084334 IC50 = 3000 nM T94879 CP6W8T 10086869 IC50 = 18500 nM T94879 CLB5S6 10087203 IC50 = 11000 nM T94879 CNA75V 10087755 IC50 = 1400 nM T94879 CJ16FV 10087963 IC50 > 1000000 nM T94879 CSP05N 10088555 IC50 = 730 nM T94879 CRW6E1 10088941 IC50 > 40000 nM T94879 C09ZNQ 10088960 IC50 = 2.6 nM T94879 C0O6MQ 10089225 IC50 = 2300 nM T94879 C13QUP 10089597 IC50 = 65000 nM T94879 CARY56 10091146 IC50 > 200000 nM T94879 CP8I5O 10093297 IC50 = 9800 nM T94879 CS4QG0 10095269 IC50 = 900 nM T94879 C61QRH 10096810 IC50 = 49000 nM T94879 CN23KJ 10105662 IC50 = 18000 nM T94879 CP3D7N 10108060 IC50 = 6000 nM T94879 C12LED 10109572 IC50 > 101000 nM T94879 CT0A4J 10113055 IC50 = 9 nM T94879 CPWL59 10113972 IC50 = 8 nM T94879 C5GRV3 10117157 IC50 = 56 nM T94879 C2PBD6 10131447 IC50 = 19300 nM T94879 C3AOI5 10138533 IC50 = 134 nM T94879 C8XPO7 10145438 Ki = 0.2 nM T94879 C4F3SH 10151707 IC50 = 1.585 nM T94879 C3H1IG 10161792 IC50 = 750 nM T94879 C89DXP 10181676 IC50 = 6 nM T94879 C5HC2X 10182563 IC50 = 52400 nM T94879 CK3TY8 10187239 IC50 = 2.089 nM T94879 CJZK81 10195399 IC50 = 1.9 nM T94879 C3GN8K 10200432 IC50 > 101000 nM T94879 CK81LJ 10203901 Ki = 4 nM T94879 CEY6F7 10205437 IC50 = 10.96 nM T94879 CLW92Y 10205894 IC50 = 65 nM T94879 CULN70 10206649 Ki = 0.31 nM T94879 C8JR4W 10221093 IC50 = 44000 nM T94879 CFGO46 10221904 IC50 = 60000 nM T94879 C8V6FE 10225063 IC50 = 2 nM T94879 CX35CL 10244508 IC50 = 6200 nM T94879 CGA50J 10244709 IC50 = 230 nM T94879 CT7RC0 10245770 IC50 = 15000 nM T94879 CC80XO 10247363 IC50 = 620 nM T94879 CP4YR0 10248176 IC50 > 1000000 nM T94879 C8G3BJ 10249105 IC50 = 3.5 nM T94879 C7MQZ1 10249183 IC50 > 1000000 nM T94879 C3AFN6 10250999 IC50 = 8300 nM T94879 CRK1U0 10252045 IC50 = 53000 nM T94879 C7GTC0 10264205 IC50 = 3020 nM T94879 C5VQL9 10264224 IC50 = 26000 nM T94879 CP70US 10267904 IC50 = 13800 nM T94879 CQ61CV 10268304 IC50 = 68400 nM T94879 C1QU2B 10268305 IC50 = 9470 nM T94879 C1VL9A 10269511 IC50 = 0.48 nM T94879 CH9C4K 10269859 IC50 = 23600 nM T94879 CR92JY 10270352 IC50 > 101000 nM T94879 C7CHR0 10270536 IC50 = 12600 nM T94879 C1VH6L 10279632 Ki = 8 nM T94879 C1FA4P 10288830 IC50 = 1.6 nM T94879 C3YO7N 10289243 IC50 = 1.288 nM T94879 CISQ36 10291967 IC50 = 63000 nM T94879 CKR74B 10292282 IC50 = 840 nM T94879 CA54BI 10294138 IC50 = 4 nM T94879 CKQ8I4 10313609 IC50 = 860 nM T94879 CUE72P 10314633 IC50 = 16 nM T94879 CJO72N 10315684 IC50 = 14 nM T94879 CIPN48 10316358 IC50 = 22000 nM T94879 C36AGZ 10321525 IC50 = 240 nM T94879 C90QZM 10324834 IC50 = 2.1 nM T94879 CRJW04 10334696 IC50 = 4000 nM T94879 C5K1LH 10336744 IC50 = 480 nM T94879 C6AQ0U 10338401 IC50 > 200000 nM T94879 C4GB5L 10338602 IC50 = 38 nM T94879 C52EPV 10339653 IC50 > 1000000 nM T94879 CMJG73 10342601 IC50 = 1200 nM T94879 CK05FV 10343476 IC50 = 68000 nM T94879 C32IUF 10344870 IC50 = 40000 nM T94879 CHZL20 10345264 IC50 = 1.6 nM T94879 CA18KO 10347662 IC50 = 20000 nM T94879 CC4W3M 10349233 IC50 = 24000 nM T94879 CQD9O7 10355498 IC50 = 6000 nM T94879 C4BL9Q 10358104 IC50 = 20000 nM T94879 CG8V6F 10358836 IC50 = 9000 nM T94879 CEIW08 10359077 IC50 = 175000 nM T94879 CP5S1A 10359273 IC50 = 165 nM T94879 C7QYK3 10359377 IC50 = 2150 nM T94879 CR35FX 10378878 IC50 = 15000 nM T94879 C2H9SE 10380126 IC50 = 4000 nM T94879 C6E5OY 10380621 IC50 = 5900 nM T94879 C5EVH3 10381520 IC50 = 380 nM T94879 C0J7OV 10382041 IC50 = 11000 nM T94879 C9IK3H 10382413 IC50 = 120 nM T94879 C52DNX 10384462 IC50 = 5500 nM T94879 CF6A1Q 10385088 IC50 > 200000 nM T94879 CZ6X9Y 10391444 IC50 = 3100 nM T94879 CQOX84 10393352 IC50 = 3.5 nM T94879 C9-APR-07 10394586 IC50 = 34000 nM T94879 CI8B3P 10401473 IC50 = 1000 nM T94879 C6E0PG 10401818 IC50 = 2000 nM T94879 C7X4EW 10402019 IC50 = 630 nM T94879 C78SRU 10403787 IC50 = 72 nM T94879 CUF0X6 10404302 IC50 > 1000000 nM T94879 C0ADP3 10404378 IC50 = 56000 nM T94879 CV3I5E 10405045 IC50 = 380 nM T94879 CP8ZV5 10408375 IC50 = 140 nM T94879 C4BF5Y 10411270 IC50 = 1.4 nM T94879 CQUE27 10413015 IC50 = 37000 nM T94879 CS7J4V 10414339 IC50 = 16 nM T94879 C0ZLB5 10423102 IC50 = 1000 nM T94879 C5ZQG3 10426854 IC50 = 5500 nM T94879 C5HMX2 10428149 IC50 = 32000 nM T94879 CB2X9W 10429802 IC50 = 110 nM T94879 CAW23H 10434818 IC50 > 1000000 nM T94879 CH76CS 10443650 IC50 = 42000 nM T94879 CBH5V4 10445800 IC50 = 24000 nM T94879 CZ8IC4 10448177 IC50 > 1000000 nM T94879 CYU38H 10448853 IC50 = 1600 nM T94879 C1RZ9E 10449000 IC50 > 1000000 nM T94879 C18EHX 10449737 IC50 = 1300 nM T94879 CU2HN6 10450290 IC50 > 200000 nM T94879 C9IF7Y 10451065 IC50 = 4.8 nM T94879 CY4O0K 10452443 IC50 = 38000 nM T94879 CI1H7F 10452463 IC50 = 0.05 nM T94879 C4LOK1 10454517 IC50 = 3600 nM T94879 CR04LJ 10456913 IC50 = 54000 nM T94879 CASV91 10466228 IC50 = 34000 nM T94879 C6IP3N 10468291 IC50 = 24000 nM T94879 C6PXC2 10471556 IC50 = 31 nM T94879 C2FYT6 10471617 IC50 = 2300 nM T94879 C2DEO3 10472374 IC50 > 200000 nM T94879 CBMI84 10473521 IC50 = 810 nM T94879 CF0I6O 10479155 IC50 = 13000 nM T94879 C5CI3G 10479468 IC50 = 53000 nM T94879 CZ92DR 10481735 IC50 = 9 nM T94879 CE2RJ7 10499713 IC50 = 420 nM T94879 C0N5LU 10504068 IC50 = 0.53 nM T94879 C71AJB 10520277 IC50 = 19 nM T94879 CSZ7L0 10520799 IC50 = 19 nM T94879 CPWU60 10524067 IC50 = 8000 nM T94879 CG1QK8 10542139 IC50 = 6200 nM T94879 C7LG4O 10543051 IC50 = 26000 nM T94879 C7K5PG 10544204 IC50 = 26 nM T94879 C0Z1CT 10546352 IC50 = 63 nM T94879 CCK5F8 10549901 IC50 = 120 nM T94879 CMK39Q 10553487 IC50 = 200 nM T94879 CQW79N 10554042 IC50 = 10000 nM T94879 CTYQ03 10565296 IC50 = 7500 nM T94879 C1DO9H 10573238 IC50 = 275 nM T94879 CI8GS1 10574005 IC50 = 590 nM T94879 CY9P5W 10575733 IC50 = 30000 nM T94879 CFY5J3 10576937 IC50 = 305 nM T94879 CYD4Z2 10592106 IC50 = 140 nM T94879 C4HVR8 10595830 IC50 = 5600 nM T94879 CRKT15 10597744 IC50 = 43 nM T94879 C71YLE 10598277 IC50 = 4 nM T94879 CJ7CU4 10603606 IC50 = 1000 nM T94879 CR9H4Z 10617782 IC50 = 4500 nM T94879 CK3GR5 10624131 IC50 = 20000 nM T94879 C25WRZ 10627119 IC50 = 9000 nM T94879 CC68NQ 10636956 IC50 = 100 nM T94879 CE57IW 10639502 IC50 = 3300 nM T94879 C0U8KD 10642598 IC50 = 10000 nM T94879 CX61NW 10642809 IC50 = 810 nM T94879 CNK65G 10646809 IC50 = 100000 nM T94879 CKNA14 10648008 IC50 = 20000 nM T94879 C32TRJ 10659857 IC50 = 240 nM T94879 C9GJ5K 10660011 IC50 = 13000 nM T94879 C8KWM5 10663015 IC50 = 34 nM T94879 CP13SC 10663562 IC50 = 80 nM T94879 COQ17R 10666144 IC50 = 9200 nM T94879 CBQ24O 10668762 IC50 = 4000 nM T94879 C1R9VY 10669652 IC50 = 110 nM T94879 CB9Y7A 10669693 IC50 = 40000 nM T94879 CWYZ15 10670833 IC50 = 2 nM T94879 C2Y5HF 10675032 IC50 = 800 nM T94879 CW12SY 10690095 IC50 = 510 nM T94879 CV6WT3 10692240 IC50 > 30000 nM T94879 C29YKI 10692613 IC50 = 1200 nM T94879 C0FPL8 10692684 IC50 = 800 nM T94879 CI6ON5 10698519 IC50 = 4000 nM T94879 C2JTX7 10715358 IC50 = 400 nM T94879 C1I8VM 10716045 IC50 = 1500 nM T94879 CDMP96 10717370 IC50 = 30000 nM T94879 CCI8R7 10729204 IC50 > 100000 nM T94879 C2P5VY 10731865 IC50 = 610 nM T94879 CSQG30 10741916 IC50 = 0.55 nM T94879 CTCS25 10753773 IC50 = 100 nM T94879 C3X8UM 10754735 IC50 = 800 nM T94879 C4EG9Z 10759241 IC50 = 19 nM T94879 CEIZ87 10761565 IC50 = 54 nM T94879 CINX82 10763354 IC50 = 20000 nM T94879 COVG15 10764868 IC50 = 120 nM T94879 C51XRM 10776762 IC50 = 2400 nM T94879 CR4O8B 10781567 IC50 = 16000 nM T94879 C7O8WB 10787783 IC50 = 180 nM T94879 CLM42P 10788651 IC50 = 20000 nM T94879 C7U2NT 10808382 IC50 = 140 nM T94879 CEI0J8 10809340 IC50 = 49 nM T94879 CDF43L 10810826 IC50 = 66 nM T94879 CTMX70 10815441 IC50 = 58000 nM T94879 CA9UW6 10816539 IC50 = 200 nM T94879 C5V1AY 10828080 IC50 = 60 nM T94879 C0SEG5 10830345 IC50 = 6000 nM T94879 CI0XH5 10833134 IC50 = 98 nM T94879 CT6VP3 10834312 IC50 = 560 nM T94879 C8HY0A 10835448 IC50 = 11 nM T94879 CZY5K8 10836947 IC50 = 600 nM T94879 CG2O1B 10836974 IC50 = 200 nM T94879 CR50XV 10841036 IC50 = 40000 nM T94879 CJ0TR9 10854527 IC50 = 100 nM T94879 CW3T1L 10863491 Ki = 154 nM T94879 C9TH7M 10863695 Ki = 1.75 nM T94879 CH0B6V 10885231 Ki = 188 nM T94879 CQ8YB7 10897309 Ki = 1.78 nM T94879 C0RTU9 10897531 EC50 = 9.5 nM T94879 CG0LM2 10907083 Ki = 0.4 nM T94879 CB6U4L 10929261 Ki = 0.47 nM T94879 CL1RW3 10929391 Ki = 0.21 nM T94879 C0BS9L 10939795 Ki = 0.71 nM T94879 C4KLI7 10951390 Ki = 1.14 nM T94879 C9UXZ6 10951441 Ki = 1.01 nM T94879 CP59RB 10968191 IC50 = 22300 nM T94879 C3GAM5 10973079 IC50 = 0.03 nM T94879 C96GWI 10983515 IC50 = 0.7 nM T94879 C84LQY 10983963 Ki = 2.59 nM T94879 CJCO78 10992580 Ki = 1.08 nM T94879 CKX30W 10994934 Ki = 0.61 nM T94879 C3EH8D 11006014 Ki = 24.7 nM T94879 CF7RW4 11016445 Ki = 2.64 nM T94879 CX1GO8 11016581 Ki = 2.71 nM T94879 CR7C1N 11017676 EC50 = 12 nM T94879 CO05WV 11024165 IC50 = 3900 nM T94879 CJMS98 11025421 Ki = 1.2 nM T94879 C3QT7I 11028215 Ki = 0.53 nM T94879 C98IUO 11039211 Ki = 0.76 nM T94879 CF6BL1 11049430 Ki = 62.8 nM T94879 C7B4MG 11071221 Ki = 1.71 nM T94879 CIO28H 11092703 Ki = 0.99 nM T94879 CG74CI 11093245 EC50 = 130 nM T94879 CW2AS4 11103879 Ki = 0.29 nM T94879 CRV32I 11114031 Ki = 3.74 nM T94879 C72TWL 11123617 Ki = 246 nM T94879 CX3N0E 11123630 Ki = 0.31 nM T94879 C24VFA 11125005 EC50 = 37 nM T94879 CL3DT7 11145432 Ki = 0.73 nM T94879 CU5C3E 11145600 Ki = 0.61 nM T94879 C3B1QP 11161553 IC50 = 21000 nM T94879 C6OH2Y 11212743 Ki = 0.22 nM T94879 CA8E0W 11212836 Ki = 0.58 nM T94879 C0FSV9 11225074 IC50 = 0.07 nM T94879 C8TD3U 11247946 IC50 = 0.14 nM T94879 C01VJK 11270159 Ki = 23.3 nM T94879 CF7R3Y 11270592 Ki = 1.06 nM T94879 C26HWL 11270869 IC50 = 0.78 nM T94879 C4R1UG 11270952 Ki = 11 nM T94879 CRZ9V8 11293623 Ki = 3.48 nM T94879 CGO29X 11318932 IC50 = 7600 nM T94879 CY9O2K 11351010 Ki = 0.35 nM T94879 CY71CZ 11351116 Ki = 4.53 nM T94879 C1YTA6 11351932 Ki = 118 nM T94879 CREQ98 11373312 IC50 = 95000 nM T94879 C4H9WX 11375723 IC50 = 320 nM T94879 CVT52P 11385644 Ki = 113 nM T94879 CPJ0Z3 11396900 Ki = 601 nM T94879 C4V6DZ 11418838 Ki = 12.5 nM T94879 C45VZC 11438405 IC50 > 16000 nM T94879 CKZ43J 11496164 IC50 = 0.08 nM T94879 CO9WX8 11497051 IC50 = 1.7 nM T94879 CS5P1N 11502459 IC50 = 2.1 nM T94879 C7S4QZ 11539946 IC50 = 1.01 nM T94879 C4ZYH9 11547485 IC50 = 2.5 nM T94879 C50BPN 11554196 IC50 = 0.65 nM T94879 CJ41RB 11560313 IC50 = 0.4 nM T94879 CJ1R6X 11568346 IC50 = 0.007 nM T94879 CL83VR 11574797 IC50 = 0.65 nM T94879 C86YZS 11575452 IC50 = 0.78 nM T94879 C53ARX 11582654 IC50 = 9.52 nM T94879 C1TOQ3 11583812 IC50 = 6.48 nM T94879 CY5JK4 11589901 IC50 = 34 nM T94879 CI6AW2 11590842 IC50 = 0.09 nM T94879 C58OXQ 11596704 IC50 = 3.3 nM T94879 CG5LT6 11605112 IC50 = 3.15 nM T94879 C7JLT3 11611915 IC50 = 0.07 nM T94879 CLU3G9 11639525 IC50 = 10 nM T94879 CO6XA4 11647832 IC50 = 0.72 nM T94879 CRK10B 11669288 IC50 = 67 nM T94879 C0B7RV 11675647 IC50 = 1.5 nM T94879 C1WV4T 11682414 IC50 = 0.5 nM T94879 C5LPU2 11690391 IC50 = 0.76 nM T94879 C5PHZ0 11710213 IC50 = 1300 nM T94879 CT69CO 11718514 IC50 = 2.6 nM T94879 C1RX0I 11720166 IC50 = 0.35 nM T94879 C7BAC0 11724504 IC50 = 4300 nM T94879 CM5T9U 11724564 IC50 = 35000 nM T94879 CNL0G1 11725859 IC50 = 10 nM T94879 C0AKJ4 11742456 IC50 > 100000 nM T94879 CA1E6R 11754694 Ki = 0.53 nM T94879 C26CKE 11754697 IC50 = 300 nM T94879 C6ERQ9 11755313 Ki = 18 nM T94879 CMP35Y 11762536 Ki = 0.15 nM T94879 C57BPZ 11763070 Ki = 1.3 nM T94879 C1K3JX 11764545 IC50 = 37000 nM T94879 CF23VJ 11775013 IC50 = 0.5012 nM T94879 C23DSJ 11782534 IC50 = 9300 nM T94879 C5EFC7 11793221 IC50 = 1000 nM T94879 CGA1F8 11794425 IC50 = 3000 nM T94879 CUM8A9 11795949 IC50 = 4300 nM T94879 C3LO2Q 11799196 IC50 = 3.1 nM T94879 C0GP6R 11812647 Ki = 0.35 nM T94879 C1J9UP 11813138 Ki = 0.52 nM T94879 CMU6W8 11826705 Ki = 1.74 nM T94879 CB4RS5 11826881 Ki = 2.09 nM T94879 C29HOL 11828590 EC50 = 44 nM T94879 CT5C0K 11849942 IC50 = 100 nM T94879 CS42FO 11849943 IC50 = 240 nM T94879 C2FZY3 11850012 IC50 = 470 nM T94879 CRY1U7 11850013 IC50 = 140 nM T94879 CVJ1X4 11850014 IC50 = 50 nM T94879 CAPF41 11850015 IC50 = 180 nM T94879 C4GQ2P 11850016 IC50 = 38 nM T94879 C4YP5D 11850079 IC50 = 40 nM T94879 C8VUW0 11850080 IC50 = 23 nM T94879 CJ6ZX9 11850081 IC50 = 8.3 nM T94879 CQ2JU9 11850082 IC50 = 79 nM T94879 CSI25Y 11850083 IC50 = 95 nM T94879 CW6D5J 11850144 IC50 = 370 nM T94879 CT9LD7 11850145 IC50 = 1500 nM T94879 C14ZXU 11850147 IC50 = 390 nM T94879 CU7X9W 11850294 IC50 = 71 nM T94879 C8ZM2F 11850366 IC50 = 220 nM T94879 CLI6G9 11850367 IC50 = 100 nM T94879 CC59AF 11850439 IC50 = 1400 nM T94879 CUK49V 11988837 Ki = 600 nM T94879 CFIO49 11988967 Ki = 1600 nM T94879 C2D0NG 11989101 Ki = 590 nM T94879 C65ABT 11989102 Ki = 1200 nM T94879 C05CLB 11992443 IC50 = 0.68 nM T94879 C0Z3KV 11992527 IC50 = 0.9 nM T94879 CXW57M 11992528 IC50 = 0.26 nM T94879 CH86SQ 11992529 IC50 = 0.11 nM T94879 CIX0V4 11992531 IC50 = 1.05 nM T94879 C7X4LC 11992631 IC50 = 0.78 nM T94879 C1B4XD 11992634 IC50 = 0.05 nM T94879 CAG1U6 11992635 IC50 = 0.1 nM T94879 CHT82G 11992739 IC50 = 0.09 nM T94879 CR4CA6 11992740 IC50 = 0.14 nM T94879 CIOU94 11992741 IC50 = 0.25 nM T94879 C95DJC 11992742 IC50 = 0.24 nM T94879 C0KM5I 11992827 IC50 = 1.1 nM T94879 CM57ID 11992831 IC50 = 0.07 nM T94879 CPX16N 11993169 IC50 = 0.07 nM T94879 C0Q4KT 11993170 IC50 = 0.04 nM T94879 C3HOV8 11993171 IC50 = 0.05 nM T94879 CZ7YR6 11993243 IC50 = 2.59 nM T94879 C4VY3X 11993244 IC50 = 0.34 nM T94879 CP4J1S 11993342 IC50 = 0.14 nM T94879 C0QZ6W 11993365 IC50 = 0.15 nM T94879 COQ5N2 11993435 IC50 = 0.43 nM T94879 C39KLP 11993437 IC50 = 1.17 nM T94879 CL8TM7 11993463 IC50 = 0.13 nM T94879 C1ZDC4 11993465 IC50 = 0.08 nM T94879 CK63SM 11993560 IC50 = 1.65 nM T94879 CIRM68 11993561 IC50 = 0.07 nM T94879 C6W2LU 11993562 IC50 = 0.13 nM T94879 C6VI5Z 12020635 Ki = 126 nM T94879 C48IYW 12020642 Ki = 24 nM T94879 CJC01W 12020645 Ki > 1000 nM T94879 CJ4H1G 12020670 Ki = 123 nM T94879 C6D0MG 12069381 IC50 = 1.4 nM T94879 C6S8LD 12355883 IC50 = 1500 nM T94879 CX0C7I 12993019 Ki = 543 nM T94879 CNR05L 12993020 Ki = 126 nM T94879 CO3G0B 12993027 Ki = 0.98 nM T94879 C09OJP 12993038 Ki = 2.07 nM T94879 CI18JL 13026433 IC50 = 1610 nM T94879 C51CKG 14583584 IC50 = 45500 nM T94879 C2ZX8H 14756622 IC50 = 1000 nM T94879 CVT43Z 15473392 IC50 = 60 nM T94879 C2RT6A 15500912 IC50 = 1.9 nM T94879 C8E4IH 15524307 IC50 = 11 nM T94879 C12BUL 15524308 IC50 = 19 nM T94879 CAC5H0 15606258 IC50 = 91000 nM T94879 C3BI9R 15951010 IC50 > 2000 nM T94879 CW6MV8 15981426 IC50 = 26 nM T94879 CYE3L9 16038477 IC50 = 2.6 nM T94879 C9OF5R 16038616 IC50 = 3.7 nM T94879 C8FJM7 16038617 IC50 = 4.5 nM T94879 C4T6CP 16038618 IC50 = 1.2 nM T94879 CIR42U 16038756 IC50 = 12 nM T94879 CF3UG1 16066664 IC50 = 0.04 nM T94879 CG1V8D 17799315 IC50 = 2.7 nM T94879 C1PZ8C 18734933 IC50 > 16000 nM T94879 C6OJI9 18796635 IC50 = 8900 nM T94879 C1FJL6 18796640 IC50 > 100000 nM T94879 CRJO82 18796649 IC50 = 4000 nM T94879 CA16YO 18796653 IC50 = 780 nM T94879 CKCM70 18796657 IC50 = 2200 nM T94879 C36LEN 18796668 IC50 = 1300 nM T94879 C0L8NR 18796689 IC50 = 1900 nM T94879 CBF8M6 18796697 IC50 = 1000 nM T94879 C3RH7V 18796719 IC50 = 11000 nM T94879 CC2WD9 18796725 IC50 > 100000 nM T94879 CNSH93 18796735 IC50 = 2000 nM T94879 CHK4Z7 18796752 IC50 = 32000 nM T94879 CNZ3I1 18796756 IC50 = 4600 nM T94879 CC1LP2 18796767 IC50 = 1000 nM T94879 C2FN9A 18796769 IC50 = 26000 nM T94879 CUE4A2 18796773 IC50 = 2000 nM T94879 C02JXD 18796791 IC50 = 1700 nM T94879 CQ8I5K 18796795 IC50 = 3500 nM T94879 CDC76R 20299686 IC50 = 26 nM T94879 CNX2D5 20646826 IC50 = 0.86 nM T94879 C36XCM 20646828 IC50 = 4.4 nM T94879 C1H2WT 20709323 IC50 = 1.8 nM T94879 C58VPG 21212519 IC50 = 2100 nM T94879 CXM8E3 21704212 IC50 = 0.79 nM T94879 CRY9Z1 21704213 IC50 = 0.32 nM T94879 CS09OZ 21704217 IC50 = 0.5 nM T94879 CH53WM 21704221 IC50 = 14 nM T94879 C7RK1W 21920272 IC50 = 5180 nM T94879 CH7N9S 21920275 IC50 = 7000 nM T94879 CV04DH 21920370 IC50 > 101000 nM T94879 C97JPF 22004355 IC50 = 6.7 nM T94879 C7DJ9E 22004357 IC50 = 2.6 nM T94879 CY6QT7 22004369 IC50 = 1.7 nM T94879 C2STP3 22004386 IC50 = 6.8 nM T94879 C7ZH2R 22004388 IC50 = 0.3 nM T94879 COM30K 22004392 IC50 = 0.7 nM T94879 C37JNS 22004412 IC50 = 0.7 nM T94879 C64YFT 22226537 IC50 = 553 nM T94879 C5G6BS 22226562 IC50 = 30 nM T94879 C70JWO 22226563 IC50 = 94 nM T94879 C8TEV5 22601583 IC50 = 0.4 nM T94879 C2FMU0 22601651 IC50 = 1.3 nM T94879 CNGD52 22744443 IC50 = 1.2 nM T94879 CMIO49 23527107 IC50 = 100 nM T94879 CZD94A 23527108 IC50 = 19 nM T94879 CW96SI 23624262 IC50 = 561 nM T94879 CXB78L 23624298 IC50 > 5000 nM T94879 C4S6VD 23654252 IC50 > 50000 nM T94879 CAJ57O 24751843 IC50 = 79000 nM T94879 CR0D6X 24751988 IC50 > 400000 nM T94879 CL79TD 24751991 IC50 = 65000 nM T94879 C51ZNR 24774842 IC50 > 5000 nM T94879 CQ19ZC 24775191 IC50 = 3500 nM T94879 C9WGI4 24802717 IC50 = 919 nM T94879 C4Y3FK 24883368 IC50 = 1.6 nM T94879 C5F6SD 24956185 IC50 = 26 nM T94879 CA9PN0 24957913 IC50 = 17 nM T94879 C6EQG2 24963293 IC50 = 0.2 nM T94879 CJ43BX 24963638 IC50 = 0.18 nM T94879 CLDO78 24963639 IC50 = 0.72 nM T94879 CG1BJ3 24965774 IC50 = 0.21 nM T94879 CDC01R 24965775 IC50 = 0.33 nM T94879 CDF34R 24966125 IC50 = 0.22 nM T94879 CNO40A 24966126 IC50 = 0.3 nM T94879 CY0G1A 24966127 IC50 = 0.23 nM T94879 CS56UN 24966128 IC50 = 1.08 nM T94879 CA25UL 24969619 IC50 = 0.31 nM T94879 C3AFU0 25093775 IC50 = 3.28 nM T94879 C93DZI 25147798 IC50 > 50000 nM T94879 CPC08B 25179287 IC50 > 50000 nM T94879 COB03R 25179478 IC50 = 40000 nM T94879 C1AV7L 30105766 IC50 = 8 nM T94879 C43UKE 42628078 IC50 = 2.4 nM T94879 CICF39 42629702 IC50 = 1850 nM T94879 CM3X9S 42629827 IC50 > 1000 nM T94879 CQN26J 42629945 IC50 = 1240 nM T94879 C6O5FX 42630062 IC50 = 2080 nM T94879 C71ZNR 42630180 IC50 = 1440 nM T94879 C4RHY0 42630191 IC50 > 5000 nM T94879 CT6RS9 42630192 IC50 = 5165 nM T94879 CYZL43 42630317 IC50 = 8780 nM T94879 CH42OZ 42630318 IC50 > 5000 nM T94879 C7X5AH 42630437 IC50 = 2050 nM T94879 CEPY38 43826154 IC50 = 200000 nM T94879 CQU19I 44180409 IC50 = 30300 nM T94879 CW8OB3 44243146 Ki = 10600 nM T94879 C19SIQ 44249786 IC50 = 14.5 nM T94879 C03DAV 44249787 IC50 = 2.3 nM T94879 CJ1GS3 44249944 IC50 = 0.9 nM T94879 CAL8X3 44264943 IC50 = 1 nM T94879 C59QCJ 44274690 IC50 = 3.89 nM T94879 C9KV6Y 44274762 IC50 = 6.457 nM T94879 CXA6Y3 44274773 IC50 = 0.61 nM T94879 CF4H9A 44274775 IC50 = 0.8913 nM T94879 CW7J4K 44274797 IC50 = 1.995 nM T94879 C9VK6M 44274798 IC50 = 5.012 nM T94879 CTP4O5 44274817 IC50 = 2.818 nM T94879 CA6J8T 44274920 IC50 = 3000 nM T94879 CV1ZA7 44280486 IC50 = 3.6 nM T94879 CG8R0W 44280487 IC50 = 4 nM T94879 CS0FX4 44280546 IC50 = 2.7 nM T94879 C05SIA 44280556 IC50 = 12.8 nM T94879 CA9KV4 44280558 IC50 = 8.4 nM T94879 CY74KE 44280614 IC50 = 19.8 nM T94879 C4RO9D 44280635 IC50 = 2.5 nM T94879 CH7W2T 44280722 IC50 = 1.2 nM T94879 CTO54N 44280723 IC50 = 0.7 nM T94879 CXRU70 44280792 IC50 = 13.2 nM T94879 CO7NV0 44280794 IC50 = 164 nM T94879 CG8I6M 44280801 IC50 = 57 nM T94879 CDQ8B2 44280847 IC50 = 1.5 nM T94879 C0N3JE 44280911 IC50 = 2 nM T94879 C3DHJ2 44280985 IC50 = 1.9 nM T94879 CA3GF6 44280994 IC50 = 127 nM T94879 CXB40D 44281036 IC50 = 28.6 nM T94879 CA1HN8 44281061 IC50 = 15.7 nM T94879 C7TKW4 44281095 IC50 = 7.1 nM T94879 CK3W1B 44281096 IC50 = 4 nM T94879 CC81DV 44281265 IC50 = 132 nM T94879 CNO94A 44281273 IC50 > 1000 nM T94879 CO1L0H 44282267 IC50 = 160 nM T94879 C79RGL 44282685 IC50 = 270 nM T94879 CK8Y4F 44286951 IC50 = 160 nM T94879 CNW8B7 44287071 IC50 = 73 nM T94879 CDHP47 44287318 IC50 = 0.6 nM T94879 C2O0JN 44307127 IC50 = 530 nM T94879 C2FW1A 44310350 IC50 = 2900 nM T94879 COP54Y 44318505 IC50 = 1.5 nM T94879 CK0N6P 44318516 IC50 = 0.95 nM T94879 C4AWN5 44318518 IC50 = 1.23 nM T94879 CP30VE 44318806 IC50 = 0.73 nM T94879 CH4T3J 44318846 IC50 = 0.7 nM T94879 CKLM51 44318862 IC50 = 150 nM T94879 CX5SO4 44320719 IC50 = 77 nM T94879 C1SI7O 44320739 IC50 = 551 nM T94879 C3TZ6O 44320740 IC50 = 105 nM T94879 CH18VT 44320762 IC50 = 135 nM T94879 C45ZJD 44320781 IC50 = 130 nM T94879 CF1DO2 44320804 IC50 = 160 nM T94879 CLBV45 44320831 IC50 = 28 nM T94879 C6RS5T 44320847 IC50 = 1360 nM T94879 CVS5D1 44320863 IC50 = 20 nM T94879 C0GM7F 44320900 IC50 = 315 nM T94879 C13WMT 44320988 IC50 = 12 nM T94879 CP78QN 44320989 IC50 = 26 nM T94879 CP34EA 44321012 IC50 = 63 nM T94879 CN8Z1I 44321013 IC50 = 24 nM T94879 CDP87G 44321026 IC50 = 3.5 nM T94879 C9G0OQ 44321064 IC50 = 19 nM T94879 CWMD23 44321111 IC50 = 5.5 nM T94879 CPEB60 44321112 IC50 = 10 nM T94879 CX9L7V 44321135 IC50 = 11 nM T94879 C51CET 44321137 IC50 = 5 nM T94879 CD0QO6 44321152 IC50 = 93 nM T94879 C69MZC 44321154 IC50 = 5420 nM T94879 CUV0W1 44321156 IC50 > 10000 nM T94879 CP71YV 44321172 IC50 = 16 nM T94879 CXNO48 44321173 IC50 > 10000 nM T94879 C7NE6Q 44321175 IC50 > 10000 nM T94879 C81WUS 44321176 IC50 = 1500 nM T94879 C4QO0A 44321178 IC50 > 10000 nM T94879 CZWA59 44321202 IC50 = 60 nM T94879 C4B1WH 44321204 IC50 = 73 nM T94879 CIAN09 44321224 IC50 = 1810 nM T94879 C86ATM 44321229 IC50 = 100 nM T94879 CR54IA 44321231 IC50 > 10000 nM T94879 C4VFQ5 44321253 IC50 = 91 nM T94879 CYVA51 44321254 IC50 > 10000 nM T94879 CUQ3R1 44321255 IC50 = 100 nM T94879 C7BM6I 44321261 IC50 = 59 nM T94879 CZ16IY 44324251 IC50 = 30000 nM T94879 CCX9Z3 44324252 IC50 = 24000 nM T94879 CG6UT1 44324296 IC50 = 20000 nM T94879 C8M4WJ 44324373 IC50 = 22000 nM T94879 CY5HZ7 44324390 IC50 = 9000 nM T94879 C5KYV6 44324391 IC50 = 8000 nM T94879 C5C4QX 44324507 IC50 = 22000 nM T94879 CNK2F8 44331802 IC50 = 270 nM T94879 CGFP09 44336826 IC50 = 0.82 nM T94879 C98VIX 44336827 IC50 = 0.69 nM T94879 C1L6SG 44336834 IC50 = 1.1 nM T94879 CH8RY1 44336844 IC50 = 1.8 nM T94879 C1AC3Z 44336847 IC50 = 0.3 nM T94879 C0NT4K 44336855 IC50 = 0.33 nM T94879 C9WLD8 44336856 IC50 = 2 nM T94879 CUME98 44336924 IC50 = 0.58 nM T94879 CM1BO3 44348247 IC50 = 32000 nM T94879 CY5L6J 44348257 IC50 = 11000 nM T94879 CD5ZW3 44348484 IC50 = 650 nM T94879 C80PGJ 44348564 IC50 = 1500 nM T94879 CY0T1M 44348625 IC50 = 9600 nM T94879 CG98RE 44358477 Ki = 3.32 nM T94879 C3H4MR 44358478 Ki = 2.49 nM T94879 CBD52Z 44358886 Ki = 4.66 nM T94879 C7LN0W 44363056 IC50 = 50 nM T94879 C71YUD 44363183 IC50 = 3000 nM T94879 CF0IB6 44377834 IC50 = 105 nM T94879 CWO45S 44377842 Ki = 145 nM T94879 C27ZVC 44377867 Ki = 132 nM T94879 C7TXQ3 44377869 Ki = 179 nM T94879 CSW1J4 44377881 Ki = 219 nM T94879 C27TDG 44377933 Ki > 100 nM T94879 C8XM3I 44377988 IC50 = 100 nM T94879 C5IOH4 44378004 IC50 = 95 nM T94879 C85XCK 44378015 Ki = 850 nM T94879 C0H7KF 44378030 Ki > 5000 nM T94879 CU29OZ 44378056 Ki = 130 nM T94879 CLV13K 44378110 Ki > 10000 nM T94879 CL3SI5 44378121 Ki = 50.6 nM T94879 CYA76O 44378142 IC50 > 10000 nM T94879 C6IOU8 44378149 Ki = 8.11 nM T94879 CBQ5W3 44378155 IC50 = 67 nM T94879 CR30BD 44378165 Ki = 32.3 nM T94879 CHL5D9 44378187 Ki = 77.5 nM T94879 CV5Y1A 44378199 Ki = 64.2 nM T94879 CT8NH9 44383851 IC50 > 10000 nM T94879 C19CRH 44383901 IC50 = 19700 nM T94879 CR9O3I 44383902 IC50 > 30000 nM T94879 CW47HV 44383906 IC50 = 17700 nM T94879 CL86MY 44383907 IC50 > 10000 nM T94879 CW63HQ 44383912 IC50 > 10000 nM T94879 CF98LG 44384286 IC50 > 10000 nM T94879 CN1WS7 44384345 IC50 = 66700 nM T94879 C01XPL 44384404 IC50 = 22700 nM T94879 CWPR87 44384405 IC50 = 2900 nM T94879 C59SDR 44384406 IC50 = 3900 nM T94879 C7WT4G 44384540 IC50 = 18200 nM T94879 C4RQB0 44384541 IC50 = 21200 nM T94879 CRZ5G8 44384546 IC50 > 100000 nM T94879 C6W4GY 44384713 IC50 = 56100 nM T94879 CKH7M8 44384714 IC50 > 30000 nM T94879 C0ZGU6 44385109 IC50 = 12100 nM T94879 CE80VB 44385244 IC50 = 1700 nM T94879 CH5GU8 44385282 IC50 = 14900 nM T94879 CL50UE 44385283 IC50 = 9700 nM T94879 CSN56E 44386916 IC50 = 3.981 nM T94879 C13HPW 44393651 IC50 > 101000 nM T94879 CJ6GB5 44393709 IC50 = 11600 nM T94879 CQP01D 44393950 IC50 = 18770 nM T94879 CU1CQ8 44394047 IC50 = 80000 nM T94879 CJYC83 44397324 IC50 = 2070 nM T94879 CZUY06 44397327 IC50 = 5620 nM T94879 CB64FY 44397328 IC50 = 1690 nM T94879 CDJ87T 44397345 IC50 = 6190 nM T94879 C5CTF6 44397346 IC50 = 140 nM T94879 C2T7BQ 44397347 IC50 = 680 nM T94879 C39VBJ 44397348 IC50 = 3350 nM T94879 CU3BF4 44397365 IC50 = 1840 nM T94879 CRTY10 44397366 IC50 = 2930 nM T94879 CYFD01 44397379 IC50 = 1510 nM T94879 C4VS1H 44397382 IC50 = 74 nM T94879 C8YCU6 44397384 IC50 = 3190 nM T94879 CQD8Z7 44397386 IC50 = 13 nM T94879 CCL9D6 44397387 IC50 = 620 nM T94879 CSAQ43 44397397 IC50 = 3190 nM T94879 C7MZ8J 44397413 IC50 = 5990 nM T94879 C8KA6R 44397415 IC50 = 920 nM T94879 CR8P4T 44397447 IC50 = 3280 nM T94879 C9TK8I 44397448 IC50 = 5150 nM T94879 CF2AP3 44397474 IC50 = 230 nM T94879 CQT12O 44397490 IC50 = 2720 nM T94879 C6FJV7 44397494 IC50 = 1280 nM T94879 CZ5QV6 44397495 IC50 = 2130 nM T94879 CAP7W0 44397504 IC50 = 1210 nM T94879 CU13ES 44397515 IC50 = 96 nM T94879 CQY79V 44397539 IC50 = 8900 nM T94879 CTAI27 44397548 IC50 = 1470 nM T94879 C98ZCS 44397556 IC50 = 270 nM T94879 CMC12S 44397573 IC50 = 6490 nM T94879 CL15YW 44397574 IC50 = 3810 nM T94879 C6GIS2 44397576 IC50 = 10000 nM T94879 C65PLD 44397577 IC50 = 4520 nM T94879 C8MFC2 44397582 IC50 = 3300 nM T94879 C3PN4D 44397598 IC50 = 790 nM T94879 CE2GZ3 44397599 IC50 = 6680 nM T94879 CY0KB5 44397600 IC50 = 2660 nM T94879 C86IAQ 44397602 IC50 = 1900 nM T94879 CR0D6I 44397603 IC50 = 8760 nM T94879 CD67XW 44397612 IC50 = 6090 nM T94879 C1ISA5 44397619 IC50 = 7820 nM T94879 CG2XI7 44397621 IC50 = 6250 nM T94879 C1HBU8 44397622 IC50 = 3160 nM T94879 CA1FG3 44397627 IC50 = 9070 nM T94879 C1FJH9 44397640 IC50 = 74 nM T94879 CV2Q1K 44397643 IC50 = 17 nM T94879 C69WZC 44397646 IC50 = 130 nM T94879 CC8Z3A 44397647 IC50 = 3680 nM T94879 C1VB8P 44397694 IC50 = 630 nM T94879 CV2M0A 44397708 IC50 = 3500 nM T94879 C8MZF1 44397709 IC50 = 4580 nM T94879 C2OA3Y 44397724 IC50 = 9460 nM T94879 CJIK26 44397727 IC50 = 320 nM T94879 CFP7S8 44397728 IC50 = 350 nM T94879 CERQ57 44397746 IC50 = 2640 nM T94879 C2PJ6R 44397748 IC50 = 10000 nM T94879 CAQD83 44397749 IC50 = 1100 nM T94879 C5GLC2 44397761 IC50 = 40 nM T94879 CUZY95 44397764 IC50 = 8620 nM T94879 CQCN29 44397781 IC50 = 770 nM T94879 C0B2YM 44397782 IC50 = 830 nM T94879 CWL0A9 44397785 IC50 = 3410 nM T94879 CSN79W 44397799 IC50 = 1800 nM T94879 C20BLM 44397801 IC50 = 1830 nM T94879 CJG87Q 44397802 IC50 = 500 nM T94879 CP1CU7 44397810 IC50 = 650 nM T94879 CI7HS1 44397811 IC50 = 6070 nM T94879 C9SQ1V 44397814 IC50 = 1450 nM T94879 CZF29N 44397816 IC50 = 190 nM T94879 CIVF18 44397836 IC50 = 890 nM T94879 CP18FI 44397837 IC50 = 2580 nM T94879 CRMN86 44397859 IC50 = 3200 nM T94879 CC7B3S 44397860 IC50 = 460 nM T94879 C01CAI 44397871 IC50 = 10000 nM T94879 C8Y0WF 44397874 IC50 = 7650 nM T94879 CJ6B1W 44397876 IC50 = 2420 nM T94879 C28ERI 44397877 IC50 = 2490 nM T94879 C6Y9XN 44397888 IC50 = 520 nM T94879 CIOM21 44397889 IC50 = 430 nM T94879 CVQ8C1 44397891 IC50 = 1240 nM T94879 CX3M5J 44397892 IC50 = 270 nM T94879 CYX72U 44397904 IC50 = 3100 nM T94879 C5JS4T 44397906 IC50 = 8910 nM T94879 CVB7K2 44397908 IC50 = 2200 nM T94879 CP8CW5 44397940 IC50 = 9430 nM T94879 CFHR09 44397941 IC50 = 9280 nM T94879 CP62TK 44397956 IC50 = 4990 nM T94879 C6UY9Z 44397957 IC50 = 4250 nM T94879 C23GTH 44397958 IC50 = 8430 nM T94879 CG36QI 44397976 IC50 = 10000 nM T94879 CDK84C 44397977 IC50 = 7560 nM T94879 CB3ZG1 44397979 IC50 = 1030 nM T94879 C4AO1D 44397980 IC50 = 9870 nM T94879 CW65CR 44397987 IC50 = 5470 nM T94879 C1DQW5 44397991 IC50 = 40 nM T94879 CP8F9A 44397992 IC50 = 8580 nM T94879 CM1ZW4 44401687 IC50 = 230 nM T94879 C0YZV7 44401690 IC50 = 33 nM T94879 C7CDY2 44401692 IC50 = 74 nM T94879 CT8R0Q 44401694 IC50 = 81 nM T94879 CDSE04 44401695 IC50 = 90 nM T94879 CB3RC6 44401705 IC50 = 60 nM T94879 CA59PR 44401708 IC50 = 81 nM T94879 CXA4D6 44401724 IC50 = 23 nM T94879 C17ODM 44401727 IC50 = 430 nM T94879 CX0AZ7 44401742 IC50 = 270 nM T94879 C3G2RU 44401767 IC50 = 350 nM T94879 C4BJ3U 44401771 IC50 = 38 nM T94879 C0F9ZD 44401772 IC50 = 2.3 nM T94879 CM45YT 44401790 IC50 = 33 nM T94879 CA1SR3 44401812 IC50 = 29 nM T94879 CN63AH 44401816 IC50 = 30 nM T94879 CVOW53 44401827 IC50 = 32 nM T94879 CVCN36 44401831 IC50 = 920 nM T94879 C59TYU 44401851 IC50 = 200 nM T94879 C78VHO 44401870 IC50 = 13000 nM T94879 CSM4X8 44401879 IC50 = 20 nM T94879 CZU4T7 44401880 IC50 = 3.3 nM T94879 C01BEI 44401886 IC50 = 100 nM T94879 CU4AR1 44401892 IC50 = 5.3 nM T94879 C14LNK 44401904 IC50 = 60 nM T94879 CVPZ92 44401905 IC50 = 28 nM T94879 C0BRH8 44401908 IC50 = 450 nM T94879 CN4T6Z 44401928 IC50 = 145 nM T94879 CV17OM 44401929 IC50 = 14 nM T94879 CK9VN7 44401931 IC50 = 320 nM T94879 C9Q1ET 44401943 IC50 = 40 nM T94879 CB98IX 44401972 IC50 = 130 nM T94879 CD51UN 44401977 IC50 = 100 nM T94879 C19QCE 44401981 IC50 = 48 nM T94879 C04BTX 44401982 IC50 = 15 nM T94879 C7MY1S 44402027 IC50 = 59 nM T94879 C6XA7P 44402060 IC50 = 3100 nM T94879 CTZ52C 44402073 IC50 = 28 nM T94879 C4P8RN 44402077 IC50 = 35 nM T94879 C6S8KA 44402114 IC50 = 40 nM T94879 CDNZ52 44402130 IC50 = 180 nM T94879 CP78NL 44402133 IC50 = 1100 nM T94879 CWVH96 44402149 IC50 = 100 nM T94879 C9BN6H 44402168 IC50 = 6.5 nM T94879 CQM65U 44402195 IC50 = 160 nM T94879 CM90NL 44402196 IC50 = 980 nM T94879 C6IY5O 44402213 IC50 = 39 nM T94879 C4O7QE 44402239 IC50 = 22 nM T94879 C4P0AC 44402278 IC50 = 75 nM T94879 C1GPC2 44402295 IC50 = 7.8 nM T94879 CCZ2E8 44438552 IC50 = 462 nM T94879 CB1C2M 44438553 IC50 = 25 nM T94879 C7RV5Q 44438554 IC50 = 20 nM T94879 CCOJ06 44438555 IC50 = 28 nM T94879 CB93RX 44438557 IC50 = 33 nM T94879 C9AO2Z 44438558 IC50 = 42 nM T94879 C50ZMB 44438560 IC50 = 5 nM T94879 C39ZMJ 44438561 IC50 = 26 nM T94879 CBQN25 44438563 IC50 = 10000 nM T94879 CJH70L 44438564 IC50 = 34 nM T94879 CE4S8J 44438565 IC50 = 51 nM T94879 CK1JU3 44459193 IC50 = 1.288 nM T94879 CZFU59 44459332 IC50 = 43 nM T94879 CJ0Q4D 44459333 IC50 = 2.2 nM T94879 CT39RH 44459469 IC50 = 2.8 nM T94879 CG4AI3 44459482 IC50 = 2.089 nM T94879 CZ6IU2 44459494 IC50 = 6.457 nM T94879 C68RBI 44459495 IC50 = 5.37 nM T94879 CNJ16Q 44459505 IC50 = 4.5 nM T94879 C0FQ1O 44459535 IC50 = 5 nM T94879 CT9R7K 44459542 IC50 = 46 nM T94879 CP97OV 44459564 IC50 = 57.54 nM T94879 C49NWP 44459572 IC50 = 550 nM T94879 C5G2JO 44459598 IC50 = 19.95 nM T94879 C8MBD9 44459599 IC50 = 158.49 nM T94879 C0W4VT 44459622 IC50 = 39.81 nM T94879 C18EJF 44459640 IC50 = 1.8 nM T94879 C7RGD3 44459641 IC50 = 2.089 nM T94879 CQ95TO 44459661 IC50 = 128.82 nM T94879 CRH7N1 44459687 IC50 = 6.31 nM T94879 C8JS2X 44459694 IC50 = 18 nM T94879 CO3F9K 44459713 IC50 = 8.3 nM T94879 CF4C3P 44459717 IC50 = 7 nM T94879 C1W5OG 44459718 IC50 = 21.88 nM T94879 C31SQM 44459720 IC50 = 2.291 nM T94879 CS17XE 44459751 IC50 = 6.761 nM T94879 C85QDR 44459752 IC50 = 13 nM T94879 CI2V6T 44459760 IC50 = 1.096 nM T94879 CJN91Z 44459761 IC50 = 0.8913 nM T94879 CQ01TE 44459776 IC50 = 3.09 nM T94879 C24BGR 44459782 IC50 = 1.514 nM T94879 CB37LV 44459783 IC50 = 6.3 nM T94879 C1V3CW 44459848 IC50 = 3.02 nM T94879 C52JOE 44459875 IC50 = 47.86 nM T94879 CZ1DJ8 44459876 IC50 = 55 nM T94879 CWXV09 44459906 IC50 = 0.3 nM T94879 CJ4L3O 44459907 IC50 = 7.943 nM T94879 CZ0DN5 44572149 IC50 > 10000 nM T94879 C6U8QW 44572150 IC50 > 10000 nM T94879 C9XD8C 44572789 IC50 = 5200 nM T94879 C72XEI 44572984 IC50 > 10000 nM T94879 CIX5Q0 44572985 IC50 > 10000 nM T94879 C7UXN8 44572986 IC50 > 10000 nM T94879 CRBQ49 44572987 IC50 = 6500 nM T94879 C0WXB4 44580020 IC50 = 1.585 nM T94879 CHA63L 44580021 IC50 = 6.31 nM T94879 CX3L1P 44587252 IC50 = 160 nM T94879 CI3K8T 44605342 IC50 = 87100 nM T94879 CV8RY3 45260952 IC50 = 3 nM T94879 CLEU14 45260983 IC50 = 12 nM T94879 C48QSY 45261659 IC50 = 1700 nM T94879 CC5Z7N 45261660 IC50 = 2300 nM T94879 C26IBG 45261674 IC50 = 5000 nM T94879 CTG0D9 45261728 IC50 = 2800 nM T94879 CS7GA3 45264997 IC50 = 760 nM T94879 C3IOB7 45265000 IC50 = 360 nM T94879 CKW39R 45267744 IC50 = 4.571 nM T94879 C9PC5S 45267756 IC50 = 223.87 nM T94879 CR7QN3 45267764 IC50 = 0.3 nM T94879 C1KTZ3 45267771 IC50 = 33.9 nM T94879 C6WLB4 45268626 IC50 = 2.5 nM T94879 CE0U3W 45268639 IC50 = 13.49 nM T94879 CR8JH9 45268646 IC50 = 33.3 nM T94879 CM8OP3 45268652 IC50 = 0.3 nM T94879 CD6A0O 45269469 IC50 = 20.3 nM T94879 CL42XG 45269481 IC50 = 3.467 nM T94879 CRWE76 45269493 IC50 = 0.4 nM T94879 CHN4F0 45269499 IC50 = 2.9 nM T94879 C6DQU1 45269515 IC50 = 534 nM T94879 CB4IO3 45269516 IC50 = 51 nM T94879 CD47UP 45270308 IC50 = 28.18 nM T94879 C4VPC6 45270320 IC50 = 1 nM T94879 CMF3T7 45270338 IC50 = 36.5 nM T94879 C1XZ4Q 45270704 IC50 = 1.21 nM T94879 C89NBL 45270705 IC50 = 1.21 nM T94879 CDWX76 45271142 IC50 = 147.91 nM T94879 C62LVH 45272043 IC50 = 52.5 nM T94879 C0AO8K 45272078 IC50 = 43 nM T94879 CN7GR1 45272848 IC50 = 1.995 nM T94879 C8RZ7H 45272849 IC50 = 2.692 nM T94879 CQ34VM 45272857 IC50 = 3 nM T94879 C5H9RX 45272874 IC50 = 22.4 nM T94879 C7X2VE 45272888 IC50 = 0.9 nM T94879 CN8G9K 45272901 IC50 = 26.7 nM T94879 C2MW1C 45272908 IC50 = 25 nM T94879 C3X7RV 45273795 IC50 = 1.288 nM T94879 C74IXB 45273827 IC50 = 0.3 nM T94879 CLZ39M 45379958 IC50 = 2.38 nM T94879 C98KFA 45486490 IC50 = 1.17 nM T94879 CGA65L 45486496 IC50 = 0.17 nM T94879 CZ8JD0 45486497 IC50 = 0.28 nM T94879 CYF73X 45486498 IC50 = 0.38 nM T94879 C86XSZ 45486501 IC50 = 0.55 nM T94879 CDYO49 45486504 IC50 = 0.06 nM T94879 CNW0I9 45486505 IC50 = 0.71 nM T94879 CWQ6Y5 45486511 IC50 = 16.3 nM T94879 CSG37U 45486513 IC50 = 2.59 nM T94879 CEX01M 45486514 IC50 = 0.32 nM T94879 C58IWJ 45486519 IC50 = 0.25 nM T94879 CE3PK0 45486527 IC50 = 0.68 nM T94879 C1ZYT9 45486549 IC50 = 2.95 nM T94879 CHE56F 45486550 IC50 = 0.34 nM T94879 C84NHX 45486564 IC50 = 0.54 nM T94879 CLMZ68 45486571 IC50 = 4 nM T94879 CB2MG1 45486572 IC50 = 0.32 nM T94879 C0MWV4 45486574 IC50 = 0.88 nM T94879 C9SI3E 45486581 IC50 = 0.36 nM T94879 C51CUF 46193118 IC50 = 640 nM T94879 CTP8R1 46193119 IC50 = 38 nM T94879 CDT4U1 46193239 IC50 = 29000 nM T94879 C0W3LE 46193243 IC50 = 100 nM T94879 CKUN01 46193244 IC50 = 88000 nM T94879 CHU8I7 46193370 IC50 = 2800 nM T94879 C7NC9V 46193371 IC50 = 60 nM T94879 CY49DB 46193372 IC50 = 320 nM T94879 CN05XT 46193373 IC50 = 41000 nM T94879 C1Q6WV 46193374 IC50 = 32000 nM T94879 C60KFT 46193375 IC50 = 50 nM T94879 C2J9IH 46193486 IC50 = 260 nM T94879 CJ86KO 46193489 IC50 = 50 nM T94879 CPYK94 46193490 IC50 = 3400 nM T94879 CHUN05 46193595 IC50 = 40 nM T94879 C5IMB2 46239424 Ki = 6400 nM T94879 CKR9P7 46239425 Ki = 8900 nM T94879 C7SLP0 46239531 Ki = 5000 nM T94879 CI1F5C 46239840 Ki > 100000 nM T94879 C26XVS 46240044 Ki = 17324 nM T94879 CC3UF9 46830325 IC50 = 0.15 nM T94879 CE4JU7 46842025 IC50 = 0.27 nM T94879 CR8JC2 46842169 IC50 = 0.27 nM T94879 CF23CG 46842171 IC50 = 0.27 nM T94879 CWY45O 46842322 IC50 = 4.1 nM T94879 CY9UB1 46842324 IC50 = 0.27 nM T94879 CVP3F6 46886964 IC50 = 0.94 nM T94879 CF49HM 46886965 IC50 = 3.92 nM T94879 CQ91ZP 46887034 IC50 = 2.96 nM T94879 CDI09L 46887035 IC50 = 0.38 nM T94879 C8X6IR 46887483 IC50 = 0.3 nM T94879 C51BJT 46887484 IC50 = 0.86 nM T94879 CB3F2M 46887522 IC50 = 1.84 nM T94879 CVX57Z 46887568 IC50 = 3.28 nM T94879 C3GW8T 46887569 IC50 = 9.79 nM T94879 C13VUK 46888519 IC50 = 0.07 nM T94879 C7G5PM 46888541 IC50 = 0.66 nM T94879 C6NIG0 46888542 IC50 = 1.4 nM T94879 CPM4S1 46888559 IC50 = 5.5 nM T94879 CV53IU 46888560 IC50 = 0.89 nM T94879 C9UY1R 46888576 IC50 = 2.5 nM T94879 CE79JU 46888577 IC50 = 1.2 nM T94879 CQ5B2F 46888578 IC50 = 2.3 nM T94879 C8ITU7 46888595 IC50 = 0.2 nM T94879 C0IQ2C 46888596 IC50 = 2 nM T94879 CS6F1J 46888597 IC50 = 0.087 nM T94879 C7B3ZY 46888631 IC50 = 0.42 nM T94879 C8FW5K 46888632 IC50 = 2.3 nM T94879 C57KWS 46888633 IC50 = 0.35 nM T94879 CS27GK 46888659 IC50 = 0.011 nM T94879 C38INP 46888660 IC50 = 0.07 nM T94879 C6WQ5Y 46888661 IC50 = 1.2 nM T94879 CZ3SO4 46888707 IC50 = 0.19 nM T94879 C02RDT 46888708 IC50 = 0.08 nM T94879 CUN72Y 46888738 IC50 = 0.05 nM T94879 C3P2IN 46933992 IC50 = 11000 nM T94879 CHA5Z0 49821469 IC50 > 1000 nM T94879 C1AYP0 49821627 IC50 > 500 nM T94879 C85AXR 49821714 IC50 > 1000 nM T94879 CZS03D 50902030 Ki > 4274 nM T94879 CH2Z1E 50902289 Ki > 7100 nM T94879 C4HJL2 50902291 Ki > 7950 nM T94879 C6A1IU 50902549 Ki > 2000 nM T94879 C3Y2AV 50903255 Ki > 2000 nM T94879 CN41YJ 50925469 IC50 = 2 nM T94879 CQ3RG5 50925470 IC50 = 7 nM T94879 C2E5JK 50940516 IC50 = 850 nM T94879 CEB5T9 50940517 IC50 = 50 nM T94879 C2C0IA 50940656 IC50 = 850 nM T94879 C4I9OJ 50940659 IC50 = 8750 nM T94879 C6F5RK 50940660 IC50 = 300 nM T94879 C9O4LE 50940680 IC50 = 590 nM T94879 CT3H4X 50940682 IC50 = 4140 nM T94879 CN4S0D 50940686 IC50 = 2310 nM T94879 CT8V2L 50940687 IC50 = 12 nM T94879 CP3G6K 50940690 IC50 = 2300 nM T94879 C7MV1Y 50940692 IC50 = 380 nM T94879 CUM0O5 50940699 IC50 = 730 nM T94879 C9IFA6 50940700 IC50 = 50 nM T94879 C7TF6Q 50940701 IC50 = 1200 nM T94879 CI3AG0 50941259 IC50 = 260 nM T94879 CCUK19 50941260 IC50 = 990 nM T94879 CY37HL 50941261 IC50 = 10 nM T94879 CC0QW5 50941262 IC50 = 1340 nM T94879 C5Q9YU 50941264 IC50 = 3300 nM T94879 C7Y8HK 50941365 IC50 = 270 nM T94879 C8WQX5 50941366 IC50 = 1110 nM T94879 C3NK7Q 50941367 IC50 = 4460 nM T94879 C3QEV9 50941368 IC50 = 290 nM T94879 CA3HQ6 50941461 IC50 = 2040 nM T94879 C8LSY4 50941462 IC50 = 190 nM T94879 C4GBV9 50941463 IC50 = 1260 nM T94879 CYL8N5 50941464 IC50 = 1350 nM T94879 C10WDU 50941465 IC50 = 260 nM T94879 C6YM0P 50941551 IC50 = 1270 nM T94879 C6R4YN 50993785 IC50 = 10000 nM T94879 C0M6XL 50993786 IC50 = 10000 nM T94879 C0OR7K 53248667 IC50 > 100000 nM T94879 CS3R1I 53248669 IC50 = 28900 nM T94879 C30RNE 53248670 IC50 = 6400 nM T94879 C1RJ7M 54580520 IC50 > 400000 nM T94879 CCXF36 54580521 IC50 = 145000 nM T94879 CZG36N 54580522 IC50 > 400000 nM T94879 C0NPM8 54580523 IC50 = 225000 nM T94879 C25VSX 54580524 IC50 > 400000 nM T94879 CBT56Y 54581676 IC50 = 5200 nM T94879 C0MN3D 54582527 IC50 = 156000 nM T94879 C6T1QX 54582528 IC50 = 350000 nM T94879 CP4N1Q 54582529 IC50 > 400000 nM T94879 CW1X3G 54583497 IC50 > 400000 nM T94879 CN96IQ 54585432 IC50 > 400000 nM T94879 CH25CO 54586393 IC50 > 400000 nM T94879 C82LED 54586394 IC50 > 400000 nM T94879 CQ1H3C 54587403 IC50 > 400000 nM T94879 C28GAC 54587404 IC50 > 400000 nM T94879 CFX89L 54587804 IC50 = 5700 nM T94879 CGF65A 54670110 IC50 > 30000 nM T94879 C90ZLC 54670399 IC50 > 30000 nM T94879 CLK61N 56587955 IC50 = 0.1 nM T94879 C4TGL7 56648496 IC50 > 1000 nM T94879 CH6C3L 56648679 IC50 > 10000 nM T94879 CCY79V 56648680 IC50 = 3110 nM T94879 CNE96P 56648857 IC50 > 10000 nM T94879 CX86AQ 56648859 IC50 > 1000 nM T94879 CPC3T4 56654131 IC50 > 10000 nM T94879 C0YD3P 56928304 IC50 > 5000 nM T94879 C8RO6A 56929788 IC50 > 1000 nM T94879 CD52CA 57391118 IC50 = 0.02 nM T94879 C7Y4BX 57391119 IC50 = 1.47 nM T94879 C4PSK2 57391120 IC50 = 0.04 nM T94879 CA1TE7 57391121 IC50 = 0.01 nM T94879 CN60KE 57391196 IC50 = 0.09 nM T94879 CM7N8I 57391197 IC50 = 0.05 nM T94879 C7VXN9 57391198 IC50 = 1.3 nM T94879 C7SC4E 57392888 IC50 = 0.44 nM T94879 CG3DF1 57392948 Ki > 10000 nM T94879 CQT1G9 57392966 IC50 = 1.38 nM T94879 CR28IN 57394623 IC50 = 0.38 nM T94879 CHZ67R 57394624 IC50 = 0.27 nM T94879 CE36TV 57394695 Ki = 24400 nM T94879 CLEY35 57396379 IC50 = 0.64 nM T94879 C7W6TP 57396380 IC50 = 0.05 nM T94879 C80CVX 57396381 IC50 = 0.01 nM T94879 C86YCU 57396469 IC50 = 0.1 nM T94879 C3M6EL 57396470 IC50 = 1.64 nM T94879 CPQ91V 57396471 IC50 = 0.22 nM T94879 CP0AB6 57396472 IC50 = 0.28 nM T94879 CNY5Z8 57398261 IC50 = 0.35 nM T94879 CH57NZ 57398879 IC50 = 15.8 nM T94879 CTYR07 57399826 IC50 = 0.04 nM T94879 CL5UP7 57401597 IC50 = 0.36 nM T94879 C37KMA 57401598 IC50 = 0.13 nM T94879 CHQ79W 57401599 IC50 = 0.02 nM T94879 CWG70K 57401600 IC50 = 0.06 nM T94879 CU5KP3 57401601 IC50 = 0.1 nM T94879 C8GD5N 57402376 IC50 = 8.2 nM T94879 CLU6J0 57403348 IC50 = 2.43 nM T94879 CD73NJ 57403349 IC50 = 0.02 nM T94879 CPA3D1 57403394 Ki = 20800 nM T94879 CEN5Z8 57403417 IC50 = 0.08 nM T94879 CY75FP 57403418 IC50 = 0.05 nM T94879 CA4KZ8 57403419 IC50 = 1.31 nM T94879 C4XMB6 58547809 IC50 > 30000 nM T94879 CEB3G9 58547814 IC50 > 30000 nM T94879 C08QVG 58547833 IC50 > 30000 nM T94879 CFVG67 58547863 IC50 > 30000 nM T94879 CYZA38 58548077 IC50 > 30000 nM T94879 CN57ZH 67426178 IC50 > 10000 nM T94879 CO8C0Z 67453423 IC50 > 2000 nM T94879 CY8J3O 68181896 IC50 = 26000 nM T94879 CUGH78 68654838 IC50 = 1000 nM T94879 CH2X0Z 69394992 IC50 = 2.884 nM T94879 CC43LF 71074083 IC50 = 437 nM T94879 C4P0XT 71092344 IC50 = 4610 nM T94879 C6DAG4 71092519 IC50 = 13900 nM T94879 C2HGI7 71153408 IC50 > 10000 nM T94879 C9GR3L 71153436 IC50 > 10000 nM T94879 CHLQ31 71530755 IC50 = 160 nM T94879 CN8KP5 71575273 IC50 = 0.27 nM T94879 C4GNJ3 71598545 IC50 > 1000 nM T94879 C0M9IA 71666277 IC50 = 21.6 nM T94879 C3O9KX 71666278 IC50 = 0.59 nM T94879 CU0M5P 71666433 IC50 = 0.19 nM T94879 CZC74T 71666437 IC50 = 1.55 nM T94879 C68SDB 71719394 IC50 = 1995.26 nM T94879 CF2W4Z 71738037 IC50 = 240 nM T94879 C95QWN 71765666 IC50 = 17 nM T94879 CZ0G2X 72165213 IC50 > 10000 nM T94879 C7XRY6 72190879 IC50 > 30000 nM T94879 CQ3GD7 72704434 Ki = 630 nM T94879 C9JE6M 75815419 IC50 = 54.3 nM T94879 C65ZBN 76323083 IC50 = 537.03 nM T94879 CZ3P5K 89706867 IC50 = 0.056 nM T94879 CF03DW 90168772 IC50 > 20000 nM T94879 CM6J9K 90168778 IC50 > 20000 nM T94879 C45QVJ 91668196 IC50 = 2300 nM T94879 C1JPD6 91844700 IC50 = 5400 nM T94879 CYQV05 92471958 IC50 = 410 nM T94879 C6TD3W 117685212 IC50 = 337 nM T94879 CVUC27 117685328 IC50 = 1.5 nM T94879 C71BEL 117824219 IC50 = 1.7 nM T94879 CFAG87 117824250 IC50 = 0.059 nM T94879 C62NZT 117824353 IC50 = 64 nM T94879 C3WT5R 117824368 IC50 = 0.29 nM T94879 CGH1Z4 117824420 IC50 = 333 nM T94879 CX12RS 117824489 IC50 = 3.8 nM T94879 CS97IT 117830474 IC50 = 45.2 nM T94879 C60ADH 117830507 IC50 = 57 nM T94879 CMJR74 117830513 IC50 = 0.32 nM T94879 CSCY01 117949009 IC50 = 9800 nM T94879 CYQ74R 118479645 IC50 > 10000 nM T94879 CVYK24 118556943 IC50 > 50000 nM T94879 CM6XW1 118724093 IC50 = 520 nM T94879 C46LFG 118724094 IC50 > 10000 nM T94879 CYM21X 118724095 IC50 = 2900 nM T94879 C4HI1Q 118729758 IC50 = 3000 nM T94879 CKBG19 118729759 IC50 = 3100 nM T94879 C8LRQ7 121370930 IC50 = 110 nM T94879 CRJE23 122185011 IC50 > 30000 nM T94879 CS6M9C 122193679 IC50 > 100000 nM T94879 CVX7U9 127029185 IC50 = 3810 nM T94879 C9OVF8 127029366 IC50 = 5.2 nM T94879 C4UR7D 127038167 IC50 > 1000 nM T94879 C4H2TJ 127038168 IC50 > 1000 nM T94879 CL9JT8 127038169 IC50 = 606 nM T94879 CJPX60 127038509 IC50 = 232 nM T94879 C26EAG 127038511 IC50 = 201 nM T94879 CTM9E4 127038512 IC50 = 279 nM T94879 C6AQ2U 127038513 IC50 = 195 nM T94879 CV1FM0 127038868 IC50 = 228 nM T94879 CADU23 127038869 IC50 = 91.6 nM T94879 CACJ46 132489333 IC50 = 5.6 nM T94879 C2P1IU 134129996 IC50 > 100000 nM T94879 CLE03O 134130328 IC50 > 100000 nM T94879 CSN6J0 134130563 IC50 > 100000 nM T94879 C0A1CZ 134131162 IC50 > 100000 nM T94879 C23CYE 134814217 IC50 = 1.41 nM T94879 CHX5W7 134908214 IC50 = 91200 nM T94879 C1QMI8 135401477 IC50 = 26.92 nM T94879 C1BA7R 135406502 IC50 = 2 nM T94879 CIC0M9 135406542 IC50 = 3 nM T94879 CL6W5K 135406554 IC50 = 5.3 nM T94879 CL6YK2 135406621 IC50 = 1.1 nM T94879 C1LG3R 135406622 IC50 = 27 nM T94879 C9S5CV 135406637 IC50 = 1.4 nM T94879 C17YXR 135406983 IC50 = 5 nM T94879 C41TDB 135413523 IC50 = 3.5 nM T94879 C5JYM4 135415122 IC50 = 3 nM T94879 CN7LX8 135415142 IC50 = 1.5 nM T94879 CJG93Q 135415214 IC50 = 3.2 nM T94879 CQOL86 135417284 IC50 = 30 nM T94879 CG96MZ 135419216 IC50 = 2 nM T94879 COD5W1 135419220 IC50 = 2000 nM T94879 CBA1Q7 135419269 IC50 = 5 nM T94879 CP4HN6 135419318 IC50 = 7 nM T94879 CCXB28 135419329 IC50 = 2 nM T94879 CL8U1V 135419421 IC50 = 3.5 nM T94879 CN1CE4 135423930 IC50 = 2 nM T94879 C1GPZ3 135423938 IC50 = 0.2 nM T94879 C7A2NS 135427992 IC50 = 7.1 nM T94879 C6UFD4 135430871 IC50 = 10 nM T94879 C1Z3WH 135430893 IC50 = 8 nM T94879 CAJU63 135430952 IC50 = 50 nM T94879 CNP87H 135433645 IC50 = 330 nM T94879 C2DAG7 135433829 IC50 = 50 nM T94879 CHD03R 135433867 IC50 = 80 nM T94879 CJ0B6N 135438524 IC50 = 9.5 nM T94879 CJ9IE8 135438525 IC50 = 21 nM T94879 C94RVJ 135438569 IC50 = 0.7 nM T94879 C1A4MY 135439488 IC50 = 100 nM T94879 C0IE4A 135443738 IC50 = 200 nM T94879 C5U1NW 135444771 IC50 = 0.48 nM T94879 CF1U2Y 135451848 IC50 = 0.52 nM T94879 C0DBS7 135452901 IC50 = 1.905 nM T94879 CFKO84 135455980 IC50 = 5.7 nM T94879 CQW8U9 135456038 IC50 = 1 nM T94879 C9LD5N 135456042 IC50 = 2.089 nM T94879 C0BQH8 135456061 IC50 = 10 nM T94879 CA83SQ 135456100 IC50 = 1 nM T94879 C4ZQ1W 135456180 IC50 = 1.3 nM T94879 CM1K9A 135456702 IC50 = 150 nM T94879 C3R8SE 135457869 IC50 = 5200 nM T94879 C6TO5S 135462289 IC50 = 4 nM T94879 CUX8S3 135462319 IC50 = 70 nM T94879 C7HC3R 135462338 IC50 = 2.5 nM T94879 CA8X3R 135462413 IC50 = 1.7 nM T94879 CY3A0S 135462886 IC50 = 2.89 nM T94879 CA9V7D 135463722 IC50 = 10 nM T94879 C4C3JV 135467743 IC50 = 6 nM T94879 CTN73W 135467948 IC50 = 1 nM T94879 CHSI34 135469671 IC50 = 10 nM T94879 CAR9X0 135474505 IC50 = 0.62 nM T94879 CADL53 135475879 IC50 = 40 nM T94879 C3IT7F 135477808 IC50 = 13 nM T94879 C9E5KR 135480166 IC50 = 20 nM T94879 CZ9HT7 135480403 IC50 = 1.7 nM T94879 CJS37E 135482260 IC50 > 101000 nM T94879 CUNL35 135484025 IC50 = 10 nM T94879 C95GLJ 135484081 IC50 = 0.69 nM T94879 CVTR78 135484097 IC50 = 1.04 nM T94879 CKP9T0 135485820 IC50 = 5.3 nM T94879 CUV8L0 135485839 IC50 = 1.1 nM T94879 C23SWA 135485841 IC50 = 1.6 nM T94879 C4ILF7 135487662 IC50 = 1.7 nM T94879 CEHK47 135487696 IC50 = 2.6 nM T94879 CEZ5P3 135487732 IC50 = 5 nM T94879 C18DSI 135489339 IC50 = 34 nM T94879 CHO1Z5 135489408 IC50 = 7 nM T94879 CBW5A9 135491781 IC50 = 3.6 nM T94879 CG82XZ 135491934 IC50 = 18.2 nM T94879 CMNE87 135491938 IC50 = 8.2 nM T94879 CLFQ43 135493551 IC50 = 3 nM T94879 C8L1NK 135494369 IC50 = 3 nM T94879 C7FM8V 135494393 IC50 = 2 nM T94879 C3D4IY 135496441 IC50 = 3 nM T94879 C2MTZ8 135497265 IC50 = 2 nM T94879 CS4NM0 135501101 IC50 = 2 nM T94879 CJ3XM0 135503009 IC50 = 14.7 nM T94879 C86THJ 135503803 IC50 = 1 nM T94879 CN4BY1 135503843 IC50 = 2 nM T94879 C7BM8D 135504134 IC50 = 70 nM T94879 CK0S3E 135505670 IC50 = 0.9 nM T94879 C4ZNY0 135505809 IC50 = 7 nM T94879 C78CIT 135505815 IC50 = 12 nM T94879 CM27YS 135506900 IC50 = 40 nM T94879 CC87SI 135510018 IC50 = 53 nM T94879 CVM2R1 135513834 IC50 = 50 nM T94879 C6GNF4 135513951 IC50 = 0.1 nM T94879 CC9N6X 135513970 IC50 = 1 nM T94879 CL1W4B 135513981 IC50 = 5 nM T94879 CYS04P 135514690 IC50 = 0.9 nM T94879 C4NSC9 135515154 IC50 = 4 nM T94879 C9IU6B 135515212 IC50 = 2.5 nM T94879 CEV79B 135515565 IC50 = 5.5 nM T94879 C0STP6 135518654 IC50 = 2.5 nM T94879 CKDH83 135518785 IC50 = 0.2 nM T94879 C8VT4S 135520162 IC50 = 6.4 nM T94879 CKD97I 135520170 IC50 = 13 nM T94879 CL0HD1 135520500 IC50 = 18 nM T94879 C5EBI4 135525517 IC50 = 44 nM T94879 CD84SI 135528161 IC50 = 35 nM T94879 CYF17I 135528172 IC50 = 3.3 nM T94879 CB6H4I 135528567 IC50 = 13 nM T94879 C6KQV1 135528758 IC50 = 5 nM T94879 CFN34H 135528775 IC50 = 4 nM T94879 CLU8A5 135529022 IC50 = 1.53 nM T94879 C6YF2L 135529725 IC50 = 8 nM T94879 CJIA83 135529861 IC50 = 20 nM T94879 CTX70E 135530119 IC50 = 2.7 nM T94879 CCM89A 135530700 IC50 = 8.5 nM T94879 C43HNQ 135531347 IC50 = 1.1 nM T94879 CV34FU 135532825 IC50 = 5.2 nM T94879 CM3GD7 135532874 IC50 = 10 nM T94879 CGWS52 135532916 IC50 = 2.47 nM T94879 CEF96L 135536692 IC50 = 30 nM T94879 CKC9M0 135536718 IC50 = 40 nM T94879 C6E0BM 135536759 IC50 = 7 nM T94879 CWRQ95 135536783 IC50 = 4 nM T94879 C1Z7AY 135536802 IC50 = 0.8 nM T94879 CSO34W 135536977 IC50 = 0.78 nM T94879 CR0VL3 135543052 IC50 = 3.7 nM T94879 C45LHQ 135543089 IC50 = 2.76 nM T94879 CX4H6D 135544114 IC50 = 9.1 nM T94879 C4ASW0 135544141 IC50 = 0.6 nM T94879 CYE4C5 135544159 IC50 = 8 nM T94879 CW53FT 135545949 IC50 = 0.31 nM T94879 CK5F9W 135546517 IC50 = 1000 nM T94879 C9VKC6 135547908 IC50 = 10.8 nM T94879 C3HTJ7 135548164 IC50 = 3 nM T94879 C2CXY7 135559102 IC50 = 17 nM T94879 C8HW0M 135565273 IC50 = 8.9 nM T94879 C6J2FV 135566412 IC50 = 110 nM T94879 CHDC83 135566745 IC50 = 1.6 nM T94879 C5S7PD 135566746 IC50 > 1000 nM T94879 C3H1QO 135566795 IC50 = 18.2 nM T94879 CN1OH0 135566796 IC50 = 77 nM T94879 C9IJK1 135566935 IC50 = 90.6 nM T94879 C7M1TE 135604959 IC50 = 5 nM T94879 C6I3HM 135678134 IC50 = 20 nM T94879 CCB89G 135723513 IC50 = 20 nM T94879 CZP1J0 135731499 IC50 = 100 nM T94879 C7VBI4 135740146 IC50 = 82 nM T94879 CIQ83H 135744761 IC50 = 300 nM T94879 C97IUH 135750162 IC50 = 37000 nM T94879 CG1AN3 135790070 IC50 = 200 nM T94879 CD5J1S 135790088 IC50 = 1.76 nM T94879 C0M1LQ 135790105 IC50 = 0.31 nM T94879 CH13EW 135832627 IC50 = 4466.84 nM T94879 C31VFB 135832642 IC50 = 4400 nM T94879 C3PO9K 135856789 IC50 = 7560 nM T94879 C7KDO8 135874585 IC50 = 150 nM T94879 C51XVI 135874586 IC50 = 60 nM T94879 CWT6F3 135890114 IC50 = 5.8 nM T94879 C1EP3X 135890118 IC50 = 6.6 nM T94879 C25PUK 135890126 IC50 = 41 nM T94879 CI4DB0 135890131 IC50 = 4.5 nM T94879 CO07ZA 135890143 IC50 = 1.23 nM T94879 CBI80F 135890150 IC50 = 1.61 nM T94879 CQ8CT6 135890151 IC50 = 4 nM T94879 C8I2XR 135890178 IC50 = 1.01 nM T94879 CTX54Z 135896326 IC50 = 1500 nM T94879 CK4X2F 135898900 IC50 = 100 nM T94879 CPNJ62 135898901 IC50 = 50 nM T94879 C43ZKU 135898902 IC50 = 320 nM T94879 CSO02I 135898910 IC50 = 200 nM T94879 C30ZQG 135898911 IC50 = 510 nM T94879 CJQ74U 135898912 IC50 = 38 nM T94879 C4TRA9 135898925 IC50 = 70 nM T94879 CM2T5C 135898926 IC50 = 140 nM T94879 CH5R6Y 135898941 IC50 = 70 nM T94879 CYJ07O 135898942 IC50 = 530 nM T94879 CR30YL 135898943 IC50 = 500 nM T94879 C0MUP5 135898944 IC50 = 310 nM T94879 CT1H3Q 135898959 IC50 = 370 nM T94879 CU3MH0 135964375 IC50 = 381 nM T94879 CI46LV 135964379 IC50 = 1050 nM T94879 C61SDR 135964388 IC50 > 10000 nM T94879 C42FTR 135964389 IC50 = 116 nM T94879 CZ5UD9 135964390 IC50 = 710 nM T94879 CUQ41O 135964394 IC50 = 2100 nM T94879 C7NRJ6 135964396 IC50 = 849 nM T94879 CY6LT4 135964400 IC50 = 4870 nM T94879 C8UT0J 135964407 IC50 = 634 nM T94879 C04IQT 135964410 IC50 = 2160 nM T94879 C98BHJ 135964418 IC50 = 3340 nM T94879 CS4FT5 135964421 IC50 = 80 nM T94879 CO51CW 135964422 IC50 = 146 nM T94879 CC3HS1 135964423 IC50 = 15 nM T94879 C7KI6V 135964424 IC50 = 1330 nM T94879 C1WB6M 135964425 IC50 = 112 nM T94879 CKSO87 135964426 IC50 = 48 nM T94879 CY24DM 135964428 IC50 = 33 nM T94879 CMYW62 135964429 IC50 = 9 nM T94879 CPL92J 135964430 IC50 = 1570 nM T94879 CLX28E 135964433 IC50 = 38 nM T94879 C6D0FX 136026515 IC50 > 10000 nM T94879 CL7BE5 136032221 IC50 = 1.7 nM T94879 C9OQ5U 136032222 IC50 = 2.1 nM T94879 C6OU3Z 136034782 IC50 = 10 nM T94879 CWPB32 136034783 IC50 = 878 nM T94879 C3KCA0 136042216 IC50 = 0.69 nM T94879 CO4FS2 136042217 IC50 = 0.75 nM T94879 C5MCV8 136042218 IC50 = 2.44 nM T94879 C0EZ4B 136042219 IC50 = 0.74 nM T94879 CX1L3V 136042220 IC50 = 0.86 nM T94879 CS32WP 136042221 IC50 = 0.26 nM T94879 C21HJT 136042222 IC50 = 1.27 nM T94879 C4DP9X 136042223 IC50 = 1.83 nM T94879 CMH5B3 136042224 IC50 = 1.36 nM T94879 CMW86G 136042225 IC50 = 1.01 nM T94879 CJ5X4O 136042226 IC50 = 1.66 nM T94879 CM1TU5 136042227 IC50 = 4.35 nM T94879 C4A6JD 136043740 IC50 = 3.1 nM T94879 CS38OR 136044186 IC50 = 0.58 nM T94879 C6LT3U 136053630 IC50 = 0.29 nM T94879 C9OTF5 136053631 IC50 = 0.28 nM T94879 C5ZIU7 136056125 IC50 = 1000 nM T94879 C70DJG 136056126 IC50 = 2.1 nM T94879 C9Q3BW 136056127 IC50 = 81.28 nM T94879 C4U1SF 136056128 IC50 = 954.99 nM T94879 CI8E5F 136056129 IC50 = 780 nM T94879 CJ43ZC 136059652 IC50 = 3 nM T94879 CZT97J 136059653 IC50 = 77 nM T94879 C2DQ4L 136059654 IC50 = 100 nM T94879 CJ1TW7 136059659 IC50 = 80 nM T94879 CE75BO 136059660 IC50 = 100 nM T94879 C58IEH 136059684 IC50 = 1.1 nM T94879 CG6E8F 136059685 IC50 = 7.7 nM T94879 C97HLB 136059686 IC50 = 5.6 nM T94879 CZQ84P 136059687 IC50 = 0.62 nM T94879 CV6PU2 136059688 IC50 = 0.89 nM T94879 C12UMG 136059728 IC50 = 370 nM T94879 C6WH2S 136078534 IC50 = 10 nM T94879 CE51KZ 136079586 IC50 = 4 nM T94879 CRP24A 136087045 IC50 = 417 nM T94879 C7SUX4 136087050 IC50 = 141 nM T94879 C8UF7G 136087052 IC50 = 3300 nM T94879 C6U2FG 136104505 IC50 = 0.18 nM T94879 CB1GP4 136104506 IC50 = 0.28 nM T94879 CIC08H 136104509 IC50 = 0.41 nM T94879 C0LRM5 136104510 IC50 = 0.34 nM T94879 CNRF74 136104512 IC50 = 0.7 nM T94879 C5LXO8 136104513 IC50 = 0.32 nM T94879 C9UK1F 136132272 IC50 = 100 nM T94879 CBO5H3 136132273 IC50 = 50 nM T94879 CPY6I0 136132274 IC50 = 500 nM T94879 CDE2S8 136132275 IC50 = 300 nM T94879 CPL26N 136132276 IC50 = 1 nM T94879 C4ZBT6 136132277 IC50 = 300 nM T94879 CJ9QG1 136132278 IC50 = 5 nM T94879 C23BTX 136132279 IC50 = 20 nM T94879 C1BFD5 136132280 IC50 = 40 nM T94879 C21FVA 136180322 IC50 = 1.5 nM T94879 C41CAD 136180323 IC50 = 1.7 nM T94879 CC42DB 136180324 IC50 = 1.9 nM T94879 CGJX71 136180325 IC50 = 3.4 nM T94879 C0W3NC 136180326 IC50 = 3.9 nM T94879 CYC9Z6 136180327 IC50 = 12 nM T94879 C5EJ0K 136180328 IC50 = 32 nM T94879 CZ1JH2 136180329 IC50 = 14 nM T94879 C9OM5D 136180330 IC50 = 2.6 nM T94879 CMF1V6 136180331 IC50 = 1.6 nM T94879 C01TYU 136180332 IC50 = 16 nM T94879 CXT68L 136180333 IC50 = 13 nM T94879 CY0T8W 136180334 IC50 = 3.3 nM T94879 C1WHX6 136197281 IC50 = 0.83 nM T94879 CQW7T0 136197286 IC50 = 0.62 nM T94879 CPA8E7 136197297 IC50 = 1.21 nM T94879 CS8TV5 136197304 IC50 = 1.7 nM T94879 COTY62 136197323 IC50 = 8.8 nM T94879 C5HIL8 136197357 IC50 = 9.6 nM T94879 CE0F5T 136197398 IC50 = 1.46 nM T94879 CK2FL9 136197415 IC50 = 5.33 nM T94879 CS16YF 136197417 IC50 = 1.86 nM T94879 CN0G6U 136197445 IC50 = 0.92 nM T94879 C8TQ7A 136217455 IC50 = 3300 nM T94879 C4JCZ7 136219297 IC50 = 272 nM T94879 CE32YG 136219298 IC50 = 21.3 nM T94879 CXOM76 136236320 IC50 = 12.6 nM T94879 C65BFU 136236321 IC50 = 58 nM T94879 C96WPH 136236322 IC50 = 8.5 nM T94879 CY2NJ1 136236323 IC50 = 4.8 nM T94879 CUS40O 136236324 IC50 = 13.7 nM T94879 CS9Z1P 136236325 IC50 = 3 nM T94879 CRZ58U 136236326 IC50 = 4.8 nM T94879 C9PIO3 136236327 IC50 = 34.3 nM T94879 CSU3J2 136236328 IC50 = 7.2 nM T94879 C5KF0V 136236329 IC50 > 2000 nM T94879 CDNI42 136236330 IC50 = 312 nM T94879 CI0M5R 136236331 IC50 = 104 nM T94879 CF43SC 136236332 IC50 = 88 nM T94879 CMGK71 136236333 IC50 = 31.5 nM T94879 C9R6HE 136236334 IC50 = 65 nM T94879 C7ZU0K 136236335 IC50 = 71 nM T94879 C2BCV9 136236336 IC50 = 450 nM T94879 CO4S8B 136236337 IC50 > 2000 nM T94879 C6N2KA 136236338 IC50 = 12.5 nM T94879 CN69OZ 136239327 IC50 = 6.2 nM T94879 C63FEW 136239328 IC50 = 29.3 nM T94879 CQZR23 136244112 IC50 = 48 nM T94879 CO9M4H 136244113 IC50 = 10.2 nM T94879 CK6GB7 136244114 IC50 = 74 nM T94879 CF5BV2 136244123 IC50 = 25.5 nM T94879 C5VT4W 136244124 IC50 = 11.1 nM T94879 CZD04T 136244125 IC50 = 2.8 nM T94879 CUQA38 136244132 IC50 = 17.4 nM T94879 CILG36 136286746 IC50 = 3 nM T94879 C39WRP 136286747 IC50 = 3 nM T94879 C7ZX5O 136286761 IC50 = 48 nM T94879 C9SV6G 136645392 IC50 = 65 nM T94879 CANQ56 136645396 IC50 = 53 nM T94879 C9TGH1 136645397 IC50 = 14 nM T94879 C1F7JV 136645401 IC50 = 144 nM T94879 C32LNQ 136645404 IC50 = 149 nM T94879 C4W0IE 136645405 IC50 = 27 nM T94879 CMIU28 136645406 IC50 = 40 nM T94879 C3K2WL 136645410 IC50 = 79 nM T94879 CC1D0X 136645415 IC50 = 20 nM T94879 C02RIK 136645417 IC50 = 12 nM T94879 C8CT0Z 136645422 IC50 = 20 nM T94879 CAWT82 136645431 IC50 = 10 nM T94879 CBZ8Q1 136645433 IC50 = 22 nM T94879 C21EJD 136645435 IC50 = 2 nM T94879 C1KTV3 136645436 IC50 = 36 nM T94879 CK1B9W 136645438 IC50 = 1 nM T94879 C6QOP7 136645441 IC50 = 7 nM T94879 CMZ71T 136645444 IC50 = 10 nM T94879 CL47WS 136645445 IC50 = 3 nM T94879 C64BZR 136645447 IC50 = 44 nM T94879 C7X1UL 136645449 IC50 = 5 nM T94879 CI9ZO7 136645454 IC50 = 13 nM T94879 CA3I8S 136645455 IC50 = 2 nM T94879 CRN16W 136645457 IC50 = 1 nM T94879 CGQ92L 136645458 IC50 = 2 nM T94879 CO5DN2 136645462 IC50 = 2 nM T94879 CRPN39 136645466 IC50 = 11 nM T94879 CL5X3G 136645467 IC50 = 3 nM T94879 C48HNY 136959539 IC50 = 74 nM T94879 C1P8ZW 136959550 IC50 = 5 nM T94879 CKU95F 136966187 IC50 = 17 nM T94879 CFRG19 136985286 IC50 = 15 nM T94879 CE7F4O 136985287 IC50 = 10 nM T94879 CFPT21 136985288 IC50 = 0.5 nM T94879 CBH5Y0 136985291 IC50 = 24 nM T94879 CDAK28 136985292 IC50 = 0.6 nM T94879 CQ9XW7 136985295 IC50 = 122 nM T94879 C1M6NW 136985296 IC50 = 31 nM T94879 CJOA28 136985302 IC50 = 3 nM T94879 C8HG0E 137051684 IC50 = 2.02 nM T94879 CANS59 137136982 IC50 = 47 nM T94879 C5AE3Q 137283418 IC50 = 19 nM T94879 C0KM1X 137288419 IC50 = 2439 nM T94879 C5QIX1 137289788 IC50 = 17 nM T94879 C5X0YR 137289866 IC50 = 7 nM T94879 CU70ZB 137289868 IC50 = 207 nM T94879 CV6AN7 137289892 IC50 = 57 nM T94879 CB14CI 137289900 IC50 = 5 nM T94879 CLY69S 137289946 IC50 = 13 nM T94879 CC5HA4 137290225 IC50 = 121 nM T94879 C4RBC7 137290234 IC50 = 4 nM T94879 CKJ6Q4 137290238 IC50 = 46 nM T94879 CR53GQ 137290273 IC50 = 34 nM T94879 C8DYG6 137290344 IC50 = 13 nM T94879 C9G3JB 137292402 IC50 = 7 nM T94879 C6MXL3 137292504 IC50 = 57 nM T94879 CAZ49O 137300702 IC50 = 4 nM T94879 CGE0J6 137300703 IC50 = 165 nM T94879 CDU43L 137300704 IC50 = 11 nM T94879 CK0QG6 137300705 IC50 = 303 nM T94879 C91IPL 137300706 IC50 = 70 nM T94879 C5UYP8 137300707 IC50 = 5 nM T94879 CHSG63 137300708 IC50 = 23 nM T94879 CX57MR 137300709 IC50 = 39 nM T94879 C54KGS 137300710 IC50 = 10 nM T94879 CQD07Z 137300711 IC50 = 20 nM T94879 C3I1CB 137300712 IC50 = 38 nM T94879 C2N9VT 137348687 IC50 > 10000 nM T94879 C14DWB 137631637 IC50 = 157510 nM T94879 CML1E3 137631792 IC50 > 100 nM T94879 CA92EX 137632005 IC50 = 31 nM T94879 C5HM3W 137632322 IC50 = 17600 nM T94879 C0SGD8 137633727 IC50 = 77 nM T94879 CTRF70 137634642 IC50 > 100 nM T94879 CO7J5T 137635211 IC50 > 100 nM T94879 CF6EZ1 137635781 IC50 > 1000000 nM T94879 CKB51U 137637339 IC50 = 100000 nM T94879 CU17GD 137637935 IC50 = 5.4 nM T94879 C8RG2S 137638853 IC50 > 100 nM T94879 CA3BX6 137639488 IC50 > 100 nM T94879 C49UCG 137642312 IC50 > 100 nM T94879 C8R1GD 137644106 IC50 > 100 nM T94879 CSQ7P5 137644148 IC50 = 16 nM T94879 CM57EI 137646989 IC50 = 3.1 nM T94879 CPLM78 137647044 IC50 = 56 nM T94879 C18JOP 137647693 IC50 = 30 nM T94879 C4V8QP 137648482 IC50 = 50000 nM T94879 CSW42J 137651273 IC50 = 50 nM T94879 CH6EC3 137653604 IC50 > 100 nM T94879 CPK1J0 137654639 IC50 > 100 nM T94879 C93WRT 137655765 IC50 > 100 nM T94879 CDQ8B5 137657724 IC50 > 100 nM T94879 CY57JX 137658794 IC50 = 21 nM T94879 C2ITK1 137660715 IC50 > 100 nM T94879 CJA7I0 137662139 IC50 = 100000 nM T94879 C6KYD7 137700754 IC50 = 4010 nM T94879 CM3UF7 137700779 IC50 > 20000 nM T94879 CPTE92 138319693 IC50 = 0.32 nM T94879 C2QLX3 138393292 IC50 > 5000 nM T94879 CF3B2O 141492937 IC50 = 0.52 nM T94879 CEK54I 141492938 IC50 = 1.2 nM T94879 CMJW70 141492939 IC50 = 3.28 nM T94879 CKB05G 141492943 IC50 = 0.53 nM T94879 CU6A0R 141492944 IC50 = 2.85 nM T94879 CW7NV6 141492945 IC50 = 0.6 nM T94879 C2NW6Y 141492955 IC50 = 0.67 nM T94879 C13PVI 141492968 IC50 = 0.6 nM T94879 C42GOU 141492970 IC50 = 26.9 nM T94879 CGNK49 141492971 IC50 = 0.82 nM T94879 CXN3U7 141492981 IC50 = 86 nM T94879 CZ0M1Y 141492988 IC50 = 1.25 nM T94879 C2T8GE 141492992 IC50 = 6.45 nM T94879 C5XTB1 141492998 IC50 = 2.5 nM T94879 C93ZIQ 141492999 IC50 = 0.39 nM T94879 CUXZ06 141493000 IC50 = 0.97 nM T94879 C7RTX9 141493002 IC50 = 3.14 nM T94879 CQV0B4 141737648 IC50 = 155 nM T94879 C0JV6Y 141737649 IC50 = 39.7 nM T94879 CSOF52 141737655 IC50 = 19.9 nM T94879 C7SRA2 141737657 IC50 = 7.02 nM T94879 CE1H7F 141737660 IC50 = 97.5 nM T94879 CA5UL8 141737663 IC50 = 61 nM T94879 C6ZA7D 141737664 IC50 = 36.9 nM T94879 CMIY07 141737666 IC50 = 21.4 nM T94879 CC61SD 141737667 IC50 = 30.3 nM T94879 C14CZJ 141737668 IC50 = 8.44 nM T94879 CTNG49 141737674 IC50 = 36.4 nM T94879 CJ38IC 141737676 IC50 = 12.7 nM T94879 C1MC5Z 141737681 IC50 = 8.68 nM T94879 CK34HF 141737682 IC50 = 50.2 nM T94879 CQCM72 141737683 IC50 = 177 nM T94879 C2MEL1 141737684 IC50 = 56.4 nM T94879 CTUL23 141737690 IC50 = 5.24 nM T94879 CMW20N 141737696 IC50 = 3.87 nM T94879 CZWD98 141737697 IC50 = 80.2 nM T94879 C7GBH6 141737698 IC50 = 52.5 nM T94879 CVQJ85 141737699 IC50 = 383 nM T94879 CO1C4S 141737703 IC50 = 27.6 nM T94879 CX9N1P 141737704 IC50 = 10.5 nM T94879 C8HEG7 141737705 IC50 = 2.92 nM T94879 C8OWX3 145964082 IC50 = 2.64 nM T94879 C0P7CN 145964738 IC50 = 3.04 nM T94879 CZ1M5C 145964966 IC50 = 1.58 nM T94879 C07GTQ 145966108 IC50 = 0.79 nM T94879 C38QXR 145966233 IC50 = 251.19 nM T94879 CUM0Y5 145968257 IC50 = 6.82 nM T94879 CO4N2T 145968939 IC50 = 2.09 nM T94879 CDHG23 145971317 IC50 = 9.63 nM T94879 CMNV65 145973708 IC50 = 1.05 nM T94879 CC7HN2 145974174 IC50 > 100000 nM T94879 CIFW03 145974279 IC50 = 0.52 nM T94879 CWM49T 145974605 IC50 = 1.63 nM T94879 C2JF3R 145974856 IC50 = 2.64 nM T94879 C8BEH3 145975382 IC50 = 2.38 nM T94879 C5C6NR 145976885 IC50 = 2.37 nM T94879 CTJ6L8 145977069 IC50 = 0.39 nM T94879 C6M5ZW 145977440 IC50 = 19.95 nM T94879 CDB1E7 145977898 IC50 = 4.38 nM T94879 CK1BR0 145978345 IC50 > 100000 nM T94879 CJD7B2 145978603 IC50 = 4.03 nM T94879 CU5VD3 145978669 IC50 = 3.82 nM T94879 C9LGT4 145979889 IC50 = 235 nM T94879 CKZ1Y6 145979895 IC50 = 170 nM T94879 C50DFR 145982956 Ki = 8 nM T94879 CKTF58 145987769 IC50 = 227 nM T94879 CJA1B0 145991631 IC50 = 81.2 nM T94879 CHJ79V 145997874 IC50 = 3390 nM T94879 CM7TX2 148279038 IC50 = 1530 nM T94879 CYPW78 155510908 IC50 = 1.55 nM T94879 C6VZ5O 155514730 IC50 = 1.69 nM T94879 CL8CU6 155521936 IC50 > 200000 nM T94879 CAUO07 155524955 IC50 = 0.54 nM T94879 CT85RG 155530589 IC50 > 200000 nM T94879 CXMU51 155537188 IC50 = 0.79 nM T94879 C1IP4D 155556194 IC50 = 3.9 nM T94879 C2DA1W 155561694 IC50 > 500000 nM T94879 CQ2R0W 155568588 IC50 > 500000 nM T94879 CV07RN 44579973 IC50 = 0.6166 nM T94879 D00REK 5712 IC50 = 31900 nM T94879 D01RLF 105078 IC50 = 794.33 nM T94879 D01TOR 667555 IC50 = 450 nM T94879 D02NWF 2573787 IC50 = 720 nM T94879 D02VRN 6442679 IC50 = 1470 nM T94879 D03BWH 44587253 IC50 = 360 nM T94879 D06NIT 135564899 IC50 = 349 nM T94879 D06TLQ 5488822 IC50 = 1700 nM T94879 D09AUL 10266864 IC50 = 260 nM T94879 D09RKU 46239428 Ki = 9700 nM T94879 D09WUP 25058047 IC50 = 74 nM T94879 D0I6XA 149784 Ki > 200000 nM T94879 D0J0CB 2753 IC50 = 7150 nM T94879 D0J7GF 780643 IC50 = 320 nM T94879 D0O3QI 10356247 IC50 = 4200 nM T94879 D0R6MT 3758 IC50 = 63000 nM T94879 D0S8AV 509245 IC50 = 16230 nM T94879 D0U8YQ 921562 IC50 = 310 nM T94879 D0V1CL 37015 IC50 = 180 nM T94879 D0V4WB 149790 IC50 > 16000 nM T94879 D0W2BI 9799499 IC50 = 700 nM T94879 D0X7SR 10246505 IC50 = 1290 nM T94879 D0YZ0L 44605341 IC50 = 12600 nM T98337 D06OMK 445643 Ki = 79 nM T98337 D02VJY 3037617 IC50 = 8520 nM T98337 D04PGB 445501 IC50 > 100000 nM T98337 CRD1T0 9811664 IC50 > 100000 nM T98337 C9IS6O 9820942 IC50 > 150000 nM T98337 CSN72K 10371065 IC50 = 8360 nM T98337 CF3GI4 10508532 Ki = 600 nM T98337 C5NB9Z 11129344 IC50 > 100000 nM T98337 CTLC58 35027274 IC50 = 3800 nM T98337 C2V6RJ 56962328 IC50 = 3900 nM T98337 CJ46RD 56962330 IC50 = 3900 nM T98337 C1BUW4 57521458 IC50 = 8500 nM T98337 CGU89M 57521460 IC50 > 100000 nM T98337 CKP31Q 57521461 IC50 = 4150 nM T98337 C7D3PN 57521557 IC50 = 15340 nM T98337 CO6T0F 57521558 IC50 = 19300 nM T98337 C2RVN0 57521777 IC50 = 4270 nM T98337 C8PY2R 57521778 IC50 = 4540 nM T98337 C0HOD9 57521879 IC50 = 4180 nM T98337 CS7B2A 57521880 IC50 = 4960 nM T98337 CGP03D 57521881 IC50 = 62800 nM T98337 C9V4QB 57521882 IC50 = 30700 nM T98337 C4C7LK 57522005 IC50 = 11600 nM T98337 C8YI0U 57522006 IC50 > 100000 nM T98337 C0KC6J 57522007 IC50 = 67100 nM T98337 CH89PN 57522008 IC50 = 28500 nM T98337 CG6TK3 57522120 IC50 = 47200 nM T98337 CWQ8J7 57522121 IC50 = 45400 nM T98337 CTCH51 57522237 IC50 = 54050 nM T98337 C8R2IJ 57522238 IC50 = 15780 nM T98337 C1PBX3 57522239 IC50 = 22600 nM T98337 CU5NP7 57522240 IC50 > 100000 nM T98337 C0P3TI 57522347 IC50 > 100000 nM T98337 C6WY9D 57522348 IC50 = 29600 nM T98337 CM7ZV1 57522349 IC50 = 88200 nM T98337 C6FQ4X 57522350 IC50 > 100000 nM T98337 CHVK79 57522455 IC50 > 100000 nM T98337 C73XQS 57522456 IC50 > 100000 nM T98337 C4OJX2 57522457 IC50 = 6200 nM T98337 CGIX69 57522458 IC50 = 16400 nM T98337 CG2SO6 57522567 IC50 = 16100 nM T98337 CR9C3F 57522569 IC50 = 27200 nM T98337 C8SP3L 57522570 IC50 > 100000 nM T98337 CQ3I7G 57522682 IC50 = 18400 nM T98337 C5QM2O 57522683 IC50 = 14700 nM T98337 CE7G2U 57522684 IC50 > 100000 nM T98337 CA4R9I 57522685 IC50 > 100000 nM T98337 C3EP9M 57522800 IC50 > 100000 nM T98337 C46EIF 57522801 IC50 = 66270 nM T98337 CC85GJ 57522802 IC50 > 50000 nM T98337 CCUW31 57522803 IC50 > 50000 nM T98337 CV58SP 57522927 IC50 = 51500 nM T98337 CT58KB 57522928 IC50 = 456 nM T98337 C95OGY 57522929 IC50 > 50000 nM T98337 CZI07G 57522930 IC50 = 2030 nM T98337 C8B9HE 57522931 IC50 = 12300 nM T98337 C7Y9SK 57523063 IC50 = 32730 nM T98337 C4S5KW 57523064 IC50 > 100000 nM T98337 CT4NB0 57523068 IC50 > 100000 nM T98337 C0NUH8 57523069 IC50 > 100000 nM T98337 C2YN0S 57523070 IC50 = 9690 nM T98337 CN1S5R 60123375 Ki = 2700 nM T98337 C2DIM5 70684253 IC50 > 100000 nM T98337 CYQH64 70684260 IC50 = 9660 nM T98337 CG5D2W 70688508 IC50 > 100000 nM T98337 CWDU09 70688522 IC50 = 9130 nM T98337 CWY7C0 70692710 IC50 = 29390 nM T98337 C5MK3W 70694725 IC50 > 100000 nM T98337 CD65LN 70694726 IC50 > 100000 nM T98337 CEZG14 70694756 IC50 > 100000 nM T98337 CU9RN3 70694757 IC50 = 2020 nM T98337 C1Q7UX 71662419 Ki > 100000 nM T98337 CR5Q3M 71662579 Ki > 100000 nM T98337 CJHR74 71662580 Ki > 100000 nM T98337 C8G3VC 71662581 Ki = 7600 nM T98337 COBA89 71662582 Ki > 100000 nM T98337 CK4E7Q 71716537 Ki = 8800 nM T98337 CWY3J5 71716538 Ki = 64800 nM T98337 CCLG13 71716539 Ki = 200 nM T98337 CUD8F9 71717141 Ki = 9800 nM T98337 C7TIC3 71717142 Ki > 100000 nM T98337 C34VNG 71717766 Ki = 1000 nM T98337 CSIY48 71717767 Ki = 51100 nM T98337 C24GAX 71718373 Ki = 1200 nM T98337 CRGS91 71718374 Ki = 2100 nM T98337 CRWB36 71718375 Ki > 100000 nM T98337 C61TIG 71718376 Ki > 100000 nM T98337 CW0T3A 71718980 Ki = 27000 nM T98337 CR9FQ3 71718981 Ki = 18100 nM T98337 CS71CH 71720178 Ki = 13900 nM T98337 C0D6ZR 71720179 Ki = 13800 nM T98337 CK36QR 71720180 Ki > 100000 nM T98337 C9TVZ3 71720822 Ki = 300 nM T98337 CUT2Y6 71720824 Ki > 100000 nM T98337 C9N7TY 71720825 Ki = 23700 nM T98337 C5EMH2 86277875 Ki = 4 nM T98337 C3XNC8 86277887 Ki = 6 nM T98337 C85VMY 91936975 Ki = 700 nM T98337 CCH84L 117967740 Ki = 4900 nM T98337 CXP8S2 117967763 Ki = 800 nM T98337 CEY28F 117967783 Ki = 1500 nM T98337 C46GRQ 117967787 Ki = 140 nM T98337 C2A8EM 117967798 Ki = 7100 nM T98337 CVP4Q3 117967801 Ki = 3400 nM T98337 CWTL26 117967814 Ki = 3400 nM T98337 C5GF3N 117967822 Ki = 3600 nM T98337 C93YQU 117967826 Ki = 62900 nM T98337 CJ26YR 117967829 Ki = 17100 nM T98337 CX51BA 117967835 Ki = 43 nM T98337 C2AF1T 117967843 Ki = 3800 nM T98337 CRCH91 117967851 Ki = 3800 nM T98337 CT3DQ5 117967872 Ki = 10000 nM T98337 C7NTU4 117967885 Ki = 19500 nM T98337 CYS70L 117967909 Ki = 13400 nM T98337 CU86WK 117967913 Ki = 4500 nM T98337 CFA74P 117967937 Ki = 6500 nM T98337 C08BKM 117967939 Ki = 12600 nM T98337 CHN52K 117967946 Ki = 1400 nM T98337 C1ZYL4 117967947 Ki = 4200 nM T98337 CA6ZJ7 117967955 Ki = 13000 nM T98337 C2QZ3D 117967964 Ki = 8700 nM T98337 C07HJM 117967978 Ki = 12000 nM T98337 CSD64M 117968002 Ki = 17800 nM T98337 CTI1X7 117968005 Ki = 1200 nM T98337 CXP8N7 117968006 Ki = 1900 nM T98337 CIS63B 117968011 Ki = 55000 nM T98337 C4LAX1 117968012 Ki = 3200 nM T98337 C58LQV 117968031 Ki = 9100 nM T98337 CF1GO9 117968050 Ki = 36700 nM T98337 CXLE07 117968053 Ki = 3100 nM T98337 CXWU20 117968117 Ki = 2800 nM T98337 CZQB61 117968118 Ki = 4300 nM T98337 C5LK3R 117968129 Ki = 345000 nM T98337 CG65FE 117968136 Ki = 2200 nM T98337 C5O7SB 117968142 Ki = 5000 nM T98337 C5EU1T 117968149 Ki = 7900 nM T98337 CEXT51 117975049 Ki = 1800 nM T98337 CNP23H 122192627 Ki = 110 nM T98337 CEMN03 122192628 Ki = 160 nM T98337 C5ZF3W 122192629 Ki = 4200 nM T98337 C6S7FW 122192630 Ki = 4100 nM T98337 C0K9LY 122192631 Ki = 2000 nM T98337 CE4H8R 122192632 Ki = 2100 nM T98337 CHF0M4 122192633 Ki = 2000 nM T98337 C4A8CV 122192634 Ki = 2500 nM T98337 CK1Y9T 122192635 Ki = 1100 nM T98337 C1MC5U 122192636 Ki = 13000 nM T98337 C1HI5B 122192637 Ki = 17000 nM T98337 C40FKQ 122192638 Ki = 9000 nM T98337 CN6C1I 122192639 Ki > 100000 nM T98337 CC0L6K 127024999 Ki = 5700 nM T98337 C0SKD7 127053468 Ki = 3900 nM T98337 C1P6LO 137642835 Ki = 24.5 nM T98337 C64OBX 145707024 Ki = 230 nM T98337 CRFO70 155516049 Ki = 7800 nM T98337 CGK3T7 155524130 Ki = 810 nM T98337 CPN64O 155525030 Ki = 2600 nM T98337 CQK12X 155526064 Ki = 330 nM T98337 CC21ES 155526980 Ki = 2000 nM T98337 C4O3HP 155529425 Ki = 280 nM T98337 CH3B0K 155535419 Ki = 1300 nM T98337 CO9CS5 155539683 Ki = 28000 nM T98337 CI78TG 155545147 Ki = 3100 nM T98337 CO7S8A 155545716 Ki = 2600 nM T98337 C4AG5E 155551666 Ki = 8200 nM T98337 CP7U4H 155552889 Ki = 2400 nM T98337 CT40BW 155554017 Ki = 490 nM T98337 CKL6H4 155562050 Ki = 650 nM T98337 C4OH7J 155564329 Ki = 1900 nM T13902 CYG60X 512874 Ki = 81.4 nM T13902 CBL1C6 10883540 EC50 = 430 nM T13902 C8C9HM 11132282 EC50 = 22 nM T13902 CB96ZX 24742075 Ki = 64.3 nM T13902 CYL7A6 24825421 EC50 = 90 nM T13902 CI38DG 24825422 EC50 = 12 nM T13902 C5T6WY 24825423 EC50 = 160 nM T13902 CB8EU6 24825424 EC50 = 100 nM T13902 CN5Q0O 24825425 EC50 = 60 nM T13902 CWQU39 24825426 EC50 = 1400 nM T13902 C5EIS2 24825427 EC50 > 10000 nM T13902 CH3YB9 24825428 EC50 = 70 nM T13902 C9NPK4 24825429 EC50 = 320 nM T13902 C7OI1S 24825430 EC50 = 2100 nM T13902 CXRQ34 24825431 EC50 = 31.62 nM T13902 C4WTY2 24825432 EC50 = 230 nM T13902 C9ZDA7 24825433 EC50 > 10000 nM T13902 CLW5C7 24825434 EC50 = 150 nM T13902 CFV48O 24825435 EC50 = 330 nM T13902 C2FKX4 24825436 EC50 = 1000 nM T13902 CV25CA 24825437 EC50 = 30 nM T13902 COM6B8 24825438 EC50 > 10000 nM T13902 CYM47L 24825439 EC50 > 10000 nM T13902 CK4AB0 24825440 EC50 > 10000 nM T13902 CN84ZX 24825441 EC50 = 1200 nM T13902 C4RS1G 52936713 EC50 = 251.19 nM T13902 CA15HU 52936816 EC50 = 398.11 nM T13902 C6BH1V 52936819 EC50 = 1000 nM T13902 CRY03J 52936822 EC50 = 2511.89 nM T13902 CWRU85 52936928 EC50 = 2511.89 nM T13902 CF7M2A 52936929 EC50 = 3162.28 nM T13902 C2GV4R 52936930 EC50 = 5011.87 nM T13902 CAT2L4 52936931 EC50 = 2511.89 nM T13902 COLN94 52936934 EC50 = 794.33 nM T13902 CR6HC7 52937033 EC50 = 100 nM T13902 C2TI8L 52937034 EC50 = 251.19 nM T13902 CCWO80 52937035 EC50 = 316.23 nM T13902 CJ6K7I 52937037 EC50 = 1995.26 nM T13902 CI4Q9R 52937137 EC50 = 1000 nM T13902 CY10CO 52937140 EC50 = 3162.28 nM T13902 C6W5GH 52937141 EC50 = 2511.89 nM T13902 CENW79 52937246 EC50 = 251.19 nM T13902 C7I0MG 52937350 EC50 = 1258.93 nM T13902 CJ3E9B 52937351 EC50 = 794.33 nM T13902 CKC03F 52937353 EC50 = 199.53 nM T13902 CO6AG4 52937354 EC50 = 1584.89 nM T13902 CM7UT9 52937355 EC50 = 158.49 nM T13902 C45YZW 52937356 EC50 = 1258.93 nM T13902 CG98BX 52937447 EC50 = 316.23 nM T13902 CX32GP 52937449 EC50 = 398.11 nM T13902 CING80 52937450 EC50 = 251.19 nM T13902 C68SHU 52937451 EC50 = 1584.89 nM T13902 CHOZ17 52937452 EC50 = 501.19 nM T13902 CL96WV 54580360 EC50 = 251.19 nM T13902 CC67DZ 126673332 Ki = 7000 nM T13902 C16CVG 138857911 EC50 = 600 nM T13902 C0NF4Q 138857912 EC50 = 15 nM T13902 CRFJ45 138857913 EC50 = 13000 nM T13902 CZ93GB 139030532 Ki = 2.1 nM T13902 CE3T1J 145984173 EC50 = 13000 nM T13902 C36QJH 145988910 EC50 = 5000 nM T13902 C97VJP 145990098 EC50 = 400 nM T13902 C0AIB6 155518824 EC50 = 40 nM T13902 C94IEB 155522101 Ki = 2400 nM T13902 CN7HV4 155522503 EC50 = 900 nM T13902 CTR04M 155524650 EC50 = 800 nM T13902 CF3P4T 155527718 EC50 = 1000 nM T13902 C7LHO4 155535510 EC50 = 2000 nM T13902 C91LUA 155539274 EC50 = 9000 nM T13902 CR8AY9 155545328 EC50 = 5000 nM T13902 CG4QF6 155551225 EC50 = 500 nM T13902 C96DYA 155554234 EC50 = 100 nM T13902 CTX5J9 155557666 EC50 = 800 nM T13902 CD8TS3 155558831 EC50 = 3000 nM T13902 CJF3I2 155564002 EC50 = 4000 nM T64213 D0CO6D 71144018 IC50 > 20000 nM T64213 C9F7YI 556143 IC50 = 10 nM T64213 CZN6S9 743974 EC50 > 125892.54 nM T64213 CEFQ61 973047 IC50 = 490 nM T64213 CO19JL 1068397 IC50 = 34 nM T64213 CSXT30 1075105 EC50 = 770 nM T64213 CE0N7K 2124297 IC50 = 4220 nM T64213 CMC2Q6 2877560 IC50 = 10000 nM T64213 CZ1L9C 2898103 IC50 = 31 nM T64213 CPS8X2 11713900 EC50 = 740 nM T64213 C7FBO1 25270198 IC50 > 100000 nM T64213 C23WVS 53361524 IC50 > 10000 nM T64213 CAW4F0 53464379 IC50 = 50 nM T64213 CC21VN 53464543 IC50 = 50 nM T64213 CU78MC 53464607 IC50 = 80 nM T64213 C7I8YR 53465062 IC50 = 10 nM T64213 C5DBC6 53465181 IC50 = 250 nM T64213 CFZQ89 59672648 IC50 = 4930 nM T64213 CIMP91 59673363 IC50 = 930 nM T64213 C0JKR9 71116078 IC50 = 16 nM T64213 CSH8F6 71116172 IC50 = 0.001 nM T64213 CH2E7C 71116460 IC50 = 1.6 nM T64213 C87JXW 71135581 IC50 = 240 nM T64213 C1TQ6W 71135583 IC50 = 140 nM T64213 C5L7HN 71135586 IC50 = 540 nM T64213 CY31NM 71135589 IC50 = 0.001 nM T64213 CSIB17 71136917 IC50 = 74 nM T64213 CN5D4T 71226967 IC50 = 49 nM T64213 CMO71T 71227359 IC50 = 1.8 nM T64213 C51APH 71227580 IC50 = 7.5 nM T64213 C4M9YA 71227675 IC50 = 4.2 nM T64213 CA8Y2J 71227691 IC50 = 14 nM T64213 CO03PX 71227697 IC50 = 1.2 nM T64213 COA09X 71227729 IC50 = 3.1 nM T64213 CXN0D7 71473867 IC50 = 0.001 nM T64213 CX51CS 71474186 IC50 = 1.7 nM T64213 C4D8YT 71474187 IC50 = 5.2 nM T64213 CWA7J3 71474188 IC50 = 1.2 nM T64213 CF50JQ 71474549 IC50 = 5.2 nM T64213 C95VNA 71474551 IC50 = 48 nM T64213 CPG0L8 71491020 IC50 = 0.5 nM T64213 CM34DA 71528444 IC50 = 200 nM T64213 CB8S7P 71528445 IC50 = 5010 nM T64213 CJMG81 71528446 IC50 = 631 nM T64213 CA7MF1 71528447 IC50 = 1000 nM T64213 C6TKZ1 71528448 IC50 = 3980 nM T64213 CCGW28 71528449 IC50 = 2510 nM T64213 C1G7SZ 71528586 IC50 = 1260 nM T64213 CB1XZ5 71528587 IC50 = 126 nM T64213 CX8V9F 71528588 IC50 = 126 nM T64213 CO91MV 71528589 IC50 = 50.1 nM T64213 C9VTG4 71528590 IC50 = 31.6 nM T64213 C15NRD 71528731 IC50 = 12.6 nM T64213 CV4L1C 71528732 IC50 = 15.8 nM T64213 C4PJA7 71528733 IC50 > 10000 nM T64213 C3OT1F 71528734 IC50 = 31.6 nM T64213 C23JVX 71528735 IC50 = 3.2 nM T64213 CW20HQ 71818431 IC50 = 6300 nM T64213 C2L7TX 71818575 IC50 = 12500 nM T64213 CAN5C1 88057277 IC50 = 60 nM T64213 CT4WJ0 90107022 IC50 = 60 nM T64213 CIE3D4 90108382 IC50 = 60 nM T64213 C1EI2P 90665449 IC50 = 2200 nM T64213 C43XPQ 90665450 IC50 = 12.9 nM T64213 CF9CT5 90665451 IC50 = 49.1 nM T64213 C6SU4X 90665452 IC50 = 49.7 nM T64213 CUQK96 90665453 IC50 = 50.5 nM T64213 CSR8D7 90665454 IC50 = 3.4 nM T64213 CXR4H8 90665455 IC50 = 3.6 nM T64213 CJCR26 90665456 IC50 = 3.8 nM T64213 C6C9KP 90665457 IC50 = 4 nM T64213 CJ06SU 91535935 IC50 = 2000 nM T64213 C8Z2ED 117848832 IC50 = 3300 nM T64213 CDNC39 118246723 IC50 > 30000 nM T64213 CMC6G4 121476731 IC50 = 2.4 nM T64213 COR6Q4 121476832 IC50 = 22 nM T64213 C5YP4M 121476835 IC50 = 290 nM T64213 C54XVT 121476884 IC50 = 37 nM T64213 C3UO2A 121476940 IC50 = 200 nM T64213 C9F6PK 121476942 IC50 > 10000 nM T64213 C3TYW2 121476950 IC50 = 240 nM T64213 CD8P1F 121476973 IC50 = 50 nM T64213 C36RBL 121476974 IC50 = 9.5 nM T64213 CZTA14 121476982 IC50 = 29 nM T64213 CL86RI 121477020 IC50 = 35 nM T64213 CK3RB5 121477188 IC50 > 10000 nM T64213 C1XNR3 121513880 IC50 = 420 nM T64213 C58IUP 122189178 IC50 = 8530 nM T64213 CT5C4U 122189179 IC50 = 390 nM T64213 C1RML6 122189180 IC50 = 710 nM T64213 C8HCS3 122189181 IC50 = 2170 nM T64213 CO8M5U 122189182 IC50 > 10000 nM T64213 CU71OA 122189183 IC50 > 10000 nM T64213 C5LZW6 122189184 IC50 = 1320 nM T64213 CDJL98 122189185 IC50 = 2110 nM T64213 CS3R2X 122189186 IC50 = 910 nM T64213 C2BCJ7 122189187 IC50 = 1280 nM T64213 CG25YT 122189188 IC50 = 800 nM T64213 C7MG6P 122189189 IC50 = 260 nM T64213 CF8H0M 122189190 IC50 = 380 nM T64213 C9U6RS 122189191 IC50 = 540 nM T64213 CGFS72 122189192 IC50 = 930 nM T64213 CJZ7Y8 132569635 IC50 = 0.22 nM T64213 CF3D1C 134132776 IC50 = 2.8 nM T64213 CL8FX6 134133585 IC50 = 2.9 nM T64213 CQ2TE9 134133674 IC50 = 6.2 nM T64213 CQ08IP 134133949 IC50 = 32 nM T64213 C2B6MJ 134134519 IC50 = 46 nM T64213 CTJF87 134134782 IC50 = 3.1 nM T64213 C6K7GU 134134874 IC50 = 19 nM T64213 C8S6CT 134135548 IC50 = 530 nM T64213 CS6U7A 134137835 IC50 = 0.57 nM T64213 CROG58 134137935 IC50 = 80 nM T64213 C8IHX2 134138693 IC50 = 11 nM T64213 CFUV82 134141361 IC50 = 4.8 nM T64213 CS1MI5 134141572 IC50 = 1.7 nM T64213 CG80PJ 134141709 IC50 = 24 nM T64213 CN7PO6 134141941 IC50 = 23 nM T64213 CSX9J5 134142444 IC50 = 4.5 nM T64213 C23GVR 134142674 IC50 = 6.7 nM T64213 C84HMG 134142778 IC50 = 32 nM T64213 CBH3N5 134142854 IC50 = 1 nM T64213 CWQL46 134143254 IC50 = 410 nM T64213 C5B0ET 134143719 IC50 = 4300 nM T64213 CT51MF 134144463 IC50 = 6.3 nM T64213 CU7Z6W 134144502 IC50 = 620 nM T64213 CC3YF9 134145287 IC50 = 24 nM T64213 CJ51TH 134145916 IC50 = 3.2 nM T64213 CFQ3K6 134146321 IC50 = 770 nM T64213 C0UAK3 134147888 IC50 = 0.9 nM T64213 CIF84U 134147900 IC50 > 10000 nM T64213 CS24KA 134151107 IC50 = 4.4 nM T64213 C7YIN4 134151570 IC50 = 8.4 nM T64213 C10JCN 134151583 IC50 = 41 nM T64213 CS9M2H 134152318 IC50 = 2.1 nM T64213 C1N0XO 134152649 IC50 = 3.2 nM T64213 CR2F9S 134153899 IC50 = 0.3 nM T64213 CWXZ15 134153919 IC50 > 10000 nM T64213 C80DVZ 134154618 IC50 = 240 nM T64213 C2DIV9 134154947 IC50 = 100 nM T64213 CM2C7B 134155100 IC50 = 1.1 nM T64213 C9S3QG 134155876 IC50 = 37 nM T64213 CU8P2F 134156601 IC50 = 0.36 nM T64213 CUN57J 134156774 IC50 = 620 nM T64213 CFM1G7 134156905 IC50 = 1.8 nM T64213 C8FP7C 134157491 IC50 = 1.9 nM T64213 C24WTD 134157985 IC50 = 6 nM T64213 C1OTG4 134367627 IC50 = 1 nM T64213 C5JV2O 134374891 IC50 = 5 nM T64213 C3TW0A 134374895 IC50 = 3.2 nM T64213 CVLH60 134374993 IC50 = 0.5 nM T64213 CF24PS 134378771 IC50 = 34 nM T64213 C47TLY 134378796 IC50 = 12 nM T64213 CPHO94 137628676 EC50 = 60 nM T64213 C4J3ZS 137632071 IC50 = 0.21 nM T64213 CQ4S0J 137635724 IC50 = 0.65 nM T64213 CG1F7Q 137636243 IC50 = 2 nM T64213 C7AN0Q 137636445 IC50 = 200 nM T64213 C6XVA3 137637570 IC50 = 2000 nM T64213 C5VWH4 137637746 IC50 = 0.62 nM T64213 CC36MB 137638989 IC50 = 500 nM T64213 CP06HM 137639654 IC50 = 2510 nM T64213 CYM4C5 137639667 IC50 = 4.2 nM T64213 C4NIF9 137639683 IC50 = 160 nM T64213 C1XGB3 137639759 IC50 = 64 nM T64213 CZWI69 137639837 IC50 = 1.3 nM T64213 C04ZQU 137640563 IC50 > 25000 nM T64213 CUW2T6 137641026 IC50 = 5010 nM T64213 CS54FI 137641584 IC50 = 40 nM T64213 CISA38 137643086 IC50 = 0.71 nM T64213 C2QP6M 137644050 IC50 = 6.8 nM T64213 CR7W9S 137645621 IC50 = 2000 nM T64213 C7L2QC 137645999 IC50 = 320 nM T64213 CWK5M9 137646962 IC50 = 2.4 nM T64213 CE56RV 137647117 IC50 = 1.3 nM T64213 CKG83O 137647502 IC50 = 0.97 nM T64213 C5G0QR 137647711 IC50 = 1.4 nM T64213 CSJI59 137647785 IC50 = 0.87 nM T64213 CTD69B 137647980 IC50 = 80 nM T64213 CRU69K 137648543 IC50 = 3980 nM T64213 C0T8DE 137649399 IC50 = 60 nM T64213 CKI1J0 137649578 IC50 = 0.39 nM T64213 C5V2WN 137649769 IC50 = 1.8 nM T64213 CJ09RP 137650429 IC50 = 3.7 nM T64213 CXKG32 137650500 IC50 = 3.9 nM T64213 CA17ES 137650754 IC50 = 6.2 nM T64213 C2X4KI 137651468 IC50 = 0.31 nM T64213 CGB1O2 137652110 IC50 = 170 nM T64213 CEC23Z 137652223 IC50 = 1000 nM T64213 CRL59S 137652676 IC50 = 0.5 nM T64213 C6G8IS 137652729 IC50 > 25000 nM T64213 CZOB89 137653593 IC50 = 50 nM T64213 COC3T7 137653869 IC50 = 0.18 nM T64213 CX3JI8 137654148 IC50 = 0.99 nM T64213 CDR68H 137655371 IC50 = 3160 nM T64213 CWH9O5 137657180 IC50 = 6.3 nM T64213 CA6PE5 137657548 IC50 = 100 nM T64213 COLZ09 137657815 IC50 = 500 nM T64213 C36QPL 137659136 IC50 = 1580 nM T64213 CSZT92 137660008 IC50 = 0.29 nM T64213 CW48BQ 137660946 IC50 = 400 nM T64213 C39HPA 137661261 IC50 = 0.19 nM T64213 C4CRB5 137661997 IC50 = 130 nM T64213 CK5GJ8 139300594 IC50 = 175 nM T64213 CYP5F2 139300600 IC50 = 53 nM T64213 CEK6B1 139300630 IC50 = 2.5 nM T64213 CJ02SL 139300726 IC50 = 100 nM T64213 CD9Q0L 139300799 IC50 = 3.8 nM T64213 CK8W0E 139300844 IC50 = 190 nM T64213 CRH14F 139300861 IC50 = 33 nM T64213 C2D9TE 141756938 IC50 = 0.5 nM T64213 CHI60S 141756971 IC50 = 2 nM T64213 C94DWA 141756975 IC50 = 2 nM T64213 C86QVB 141756989 IC50 = 3.2 nM T64213 C9RI2N 141757015 IC50 = 7.9 nM T64213 C53UZY 141757055 IC50 = 0.3 nM T64213 CD05NR 145952261 IC50 = 40 nM T64213 C7Q8VT 145953322 IC50 = 150 nM T64213 C4RD5Z 145954475 IC50 = 1500 nM T64213 CVF6M0 145954552 IC50 = 6300 nM T64213 CE06FU 145955149 IC50 = 50 nM T64213 CCWK87 145956421 IC50 = 150 nM T64213 C5M7JA 145957240 IC50 = 100 nM T64213 CL75MA 145957491 IC50 = 200 nM T64213 CJ1OZ4 145972905 IC50 = 320 nM T64213 C9DO8U 145974540 IC50 = 1000 nM T64213 C7Y6WX 155510800 IC50 = 240 nM T64213 C5ESP7 155512077 EC50 = 10000 nM T64213 CT7JO0 155514099 EC50 = 920 nM T64213 C6TVW5 155515017 IC50 = 290 nM T64213 CJ97CN 155515493 IC50 = 20 nM T64213 CS6UN3 155517309 IC50 = 159 nM T64213 CZ1O0S 155518646 IC50 = 84 nM T64213 CW4J8P 155519095 EC50 > 30000 nM T64213 CE4FD0 155520787 EC50 = 125 nM T64213 CW34OZ 155520969 EC50 = 4700 nM T64213 CZVJ89 155521210 IC50 = 340 nM T64213 CW9RA8 155521362 IC50 = 1700 nM T64213 CQ10LO 155522731 IC50 = 631 nM T64213 CJ2EU3 155523773 EC50 = 1444 nM T64213 C65AUT 155525085 EC50 = 870 nM T64213 CI10UW 155526744 IC50 > 10000 nM T64213 CH0QA6 155526974 IC50 = 240 nM T64213 CT18PY 155527522 IC50 = 0.85 nM T64213 C6IUQ5 155527836 IC50 = 1.9 nM T64213 C1BL2M 155529532 IC50 = 1900 nM T64213 C4FC0I 155529667 IC50 = 310 nM T64213 C9IGK8 155529802 IC50 = 81 nM T64213 CE09AV 155530174 IC50 = 3600 nM T64213 C7CB1N 155530853 IC50 = 3.3 nM T64213 C8QC3R 155530856 IC50 = 32 nM T64213 CF56BN 155531068 EC50 = 12200 nM T64213 CHM17E 155531143 EC50 = 663 nM T64213 C7XU4P 155532190 IC50 = 3800 nM T64213 C5J8SU 155532311 IC50 = 20 nM T64213 C70HOZ 155532522 IC50 = 99 nM T64213 C4X1GY 155532905 IC50 = 25 nM T64213 C72WUI 155533369 IC50 = 1585 nM T64213 C0BH7X 155534103 IC50 = 880 nM T64213 C65PYC 155535183 IC50 > 25000 nM T64213 C36TSC 155536738 IC50 = 40 nM T64213 CP2UV1 155536845 EC50 = 200 nM T64213 C8EQ5U 155538902 IC50 = 45900 nM T64213 CVDF60 155539376 IC50 = 2.5 nM T64213 CBS40J 155540061 EC50 = 910 nM T64213 CW2V3F 155540455 IC50 = 3.5 nM T64213 CH69QA 155541913 IC50 = 22 nM T64213 CAD76Y 155542105 IC50 = 78 nM T64213 CU7I5K 155543594 IC50 = 5200 nM T64213 CPA6K3 155544013 IC50 = 30 nM T64213 CZAM13 155546455 IC50 = 15 nM T64213 C8V5ZC 155546887 IC50 = 730 nM T64213 C7VT8U 155547220 IC50 = 50 nM T64213 C6NTP5 155547945 IC50 = 63 nM T64213 C3W4YN 155548551 IC50 = 1.5 nM T64213 C5MFS0 155549146 IC50 = 11 nM T64213 CJCO06 155550779 IC50 = 820 nM T64213 CU62IK 155551656 EC50 = 670 nM T64213 CJ4FZ7 155554984 IC50 = 51 nM T64213 C8YN0J 155555089 IC50 = 830 nM T64213 CP4KU2 155555477 IC50 = 1800 nM T64213 CGM04A 155555681 IC50 = 144 nM T64213 C2YO0Z 155556366 EC50 > 30000 nM T64213 CWQ6L8 155558548 EC50 = 280 nM T64213 C2N0DM 155562973 IC50 = 310 nM T64213 C74QRJ 155563663 IC50 = 11 nM T64213 CN6ZL9 155564707 IC50 = 1.2 nM T64213 CB6G1D 155565343 IC50 = 84 nM T64213 CVRC68 155566379 EC50 = 2060 nM T64213 C2GP3W 155567128 IC50 = 86 nM T64213 CQ1PK4 155567723 IC50 = 120 nM T64213 CU7ZA1 155568064 IC50 = 96 nM T64213 CU1QT3 155568605 EC50 = 1180 nM T64213 D03HJW 23630211 EC50 = 49 nM T64213 D03LVL 53464483 IC50 = 40 nM T64213 D03OLU 3601086 IC50 = 2300 nM T64213 D0A1UL 49783953 IC50 > 10000 nM T64213 D0B1QM 2742550 IC50 = 29 nM T64213 D0D6MC 1150897 IC50 > 10000 nM T88531 CZN6S9 743974 EC50 > 50118.72 nM T88531 CW2C5H 3007855 EC50 = 3.6 nM T88531 CS6N0M 3395869 EC50 = 81 nM T88531 CR6C3X 3722317 EC50 = 200 nM T88531 CA8G7X 5407221 EC50 = 1100 nM T88531 C4G1TP 9586016 EC50 = 750 nM T88531 CV03NI 76313672 EC50 = 190 nM T88531 C9WES7 76317176 EC50 = 3100 nM T88531 CTQ0J8 76331797 EC50 = 310 nM T88531 C0V5EC 91826086 EC50 = 0.06 nM T88531 CV4CY0 118716400 EC50 = 202 nM T88531 C1B0TF 118716401 EC50 = 11 nM T88531 CW8AH5 118716402 EC50 = 164 nM T88531 C94MPI 118716403 EC50 = 5000 nM T88531 CV8ZA2 118716404 EC50 = 2204 nM T88531 CDP1U2 118716405 EC50 = 600 nM T88531 CZM50U 118716406 EC50 = 22000 nM T88531 C28OWZ 118716407 EC50 > 25000 nM T88531 C4O2IK 118716408 EC50 = 73 nM T88531 CZE4D9 118716409 EC50 = 11 nM T88531 CVX96A 118716410 EC50 = 15 nM T88531 C0T9RJ 118716411 EC50 = 87 nM T88531 CVT81A 118716412 EC50 = 1181 nM T88531 CW45UK 118716413 EC50 = 60 nM T88531 C5LB7A 118716414 EC50 = 25 nM T88531 CKJS72 118716415 EC50 = 13 nM T88531 C4TEZ0 118716416 EC50 = 36 nM T88531 CD02BX 118716417 EC50 = 0.18 nM T88531 C7TYG0 118716418 EC50 = 0.55 nM T88531 C5OHS8 118716419 EC50 = 30 nM T88531 C2JH5T 118716420 EC50 = 0.35 nM T88531 CD7E4C 135411687 EC50 = 240 nM T88531 CSP2W4 135634901 EC50 = 9 nM T88531 CJG4B1 135634945 EC50 = 18 nM T88531 C1APT5 135634948 EC50 = 460 nM T88531 C4U8WO 135893117 EC50 > 10000 nM T88531 CY17RE 137631764 EC50 = 4 nM T88531 C3V4NZ 137633165 EC50 = 3000 nM T88531 C9ZLJ0 137633277 EC50 = 10 nM T88531 C9P1BR 137635316 EC50 = 4 nM T88531 C4UC1Z 137636773 EC50 = 4 nM T88531 CW57DU 137636882 EC50 = 3 nM T88531 CB87SI 137637255 EC50 = 6 nM T88531 CPM64D 137638361 EC50 = 3 nM T88531 CQM3N5 137639471 EC50 = 1 nM T88531 C3D6TJ 137641632 EC50 = 340 nM T88531 CP15JM 137642799 EC50 = 32 nM T88531 C3LHM1 137643474 EC50 = 2 nM T88531 CJ6ZG0 137644264 EC50 = 5 nM T88531 C9B5HG 137644326 EC50 = 10 nM T88531 C7QE2R 137644868 EC50 = 8 nM T88531 CI5B1O 137645445 EC50 = 4 nM T88531 CUYQ58 137646005 EC50 = 4 nM T88531 C5HT9J 137647882 EC50 = 5 nM T88531 C1X6WC 137648191 EC50 = 2 nM T88531 CA5EG0 137648315 EC50 = 5 nM T88531 CNXI18 137649835 EC50 = 16 nM T88531 CUK3N6 137650161 EC50 = 7 nM T88531 C2CNJ7 137654391 EC50 = 4 nM T88531 CJM8Y0 137656189 EC50 = 16 nM T88531 CQ7MO9 137657224 EC50 = 2 nM T88531 C83CYS 137657821 EC50 = 5 nM T88531 C6JL1V 137658295 EC50 = 8 nM T88531 CI5KZ6 137658694 EC50 = 3 nM T88531 CNXE98 137660912 EC50 = 3 nM T88531 CF1DS8 137661197 EC50 = 1.5 nM T88531 CWQ13R 137661496 EC50 = 18 nM T88531 CX1EB4 137662043 EC50 = 3 nM T88531 D0H4UN 73211886 EC50 = 56 nM T88531 D0V6KN 86277841 EC50 = 0.8 nM T73725 D09JEJ 24748573 IC50 = 3.8 nM T73725 D0E3TC 44259 IC50 = 5.52 nM T73725 D03BNU 59604787 IC50 > 10000 nM T73725 D05BVP 3232621 IC50 = 1902 nM T73725 D09CDR 77105816 IC50 = 80 nM T73725 D0CC7E 77105818 IC50 = 150 nM T73725 D0JQ0Z 46916176 IC50 = 584 nM T73725 D0PO8N 117881270 IC50 = 15 nM T73725 CU80LI 3233012 IC50 = 692 nM T73725 CW4C3P 3235048 IC50 > 10000 nM T73725 CGAT36 5327151 IC50 = 498 nM T73725 CR3BS0 12248905 IC50 = 1100 nM T73725 C5VPH9 16129448 IC50 = 211 nM T73725 C7YG1N 24759534 IC50 < 10 nM T73725 CGLQ20 44223952 IC50 = 1327 nM T73725 CR6VH2 44223953 IC50 = 2163 nM T73725 C2IBW0 44223954 IC50 = 2219 nM T73725 CS3Q2Y 44223955 IC50 = 1810 nM T73725 C5M1UN 44223957 IC50 = 3118 nM T73725 CK8G1T 44223965 IC50 = 801 nM T73725 CJ8KD4 44223966 IC50 = 651 nM T73725 CCW0V4 44223967 IC50 = 3594 nM T73725 CF78WD 44223968 IC50 > 10000 nM T73725 CNE30X 44223970 IC50 = 186 nM T73725 CYR45S 44223971 IC50 = 589 nM T73725 CLZ62P 44223973 IC50 = 173 nM T73725 CIXB09 44223974 IC50 = 2725 nM T73725 C2OBX8 44223977 IC50 = 877 nM T73725 C3VRO9 44557921 IC50 > 10000 nM T73725 C3JBN1 44968184 IC50 = 962 nM T73725 CYW79D 44968186 IC50 = 447 nM T73725 C5OYK3 44968199 IC50 = 8510 nM T73725 C2T0EM 44968221 IC50 = 6181 nM T73725 C8NA2J 44968224 IC50 = 1209 nM T73725 CR8DC5 44968225 IC50 = 3331 nM T73725 CV19YK 44968230 IC50 = 889 nM T73725 CD4ZN1 44968231 IC50 = 1648 nM T73725 C16QFN 46172966 IC50 > 10000 nM T73725 CB32ET 46172972 IC50 > 10000 nM T73725 CN26HW 46172980 IC50 = 409 nM T73725 CGH05O 46172984 IC50 = 1092 nM T73725 CLS29B 46872626 IC50 > 10000 nM T73725 C15EJK 46916169 IC50 = 1361 nM T73725 CHG8C4 46916170 IC50 = 414 nM T73725 CI56BA 46916172 IC50 = 195 nM T73725 CZ5DJ4 46916177 IC50 = 301 nM T73725 CXK37B 46916178 IC50 = 1055 nM T73725 CL1GW0 46916179 IC50 = 486 nM T73725 CZ6DK4 46916182 IC50 = 882 nM T73725 CCUG10 46926515 IC50 = 345 nM T73725 C9NC6W 46926516 IC50 = 52 nM T73725 CZ1D2A 46926518 IC50 = 60 nM T73725 C7S6HT 46926519 IC50 = 39 nM T73725 CG1K5A 46926520 IC50 = 1557 nM T73725 CVF48X 46926521 IC50 = 259 nM T73725 C4ULH5 46926522 IC50 = 41 nM T73725 CPE98Z 46926523 IC50 = 20 nM T73725 C6WLX1 46926524 IC50 = 8791 nM T73725 C61LUI 46926526 IC50 > 10000 nM T73725 C0IVD1 46926527 IC50 = 30 nM T73725 CAYI59 49795862 IC50 = 429 nM T73725 C1UQN4 49795863 IC50 = 238 nM T73725 CU8OC0 49795864 IC50 = 1903 nM T73725 C7T5HW 49795865 IC50 = 462 nM T73725 C6N8EY 49795866 IC50 = 190 nM T73725 C7XS1Z 49795867 IC50 = 665 nM T73725 C5EWG8 49855158 IC50 = 4600 nM T73725 CS6N8Z 54581884 IC50 = 8480 nM T73725 CT6XL0 57466811 IC50 = 117 nM T73725 CXJ63M 59603829 IC50 < 10 nM T73725 CQEU96 59603842 IC50 = 14 nM T73725 CW9AE7 60034150 IC50 = 190 nM T73725 C37NKO 67129970 IC50 = 6440 nM T73725 CK80LJ 67130050 IC50 > 10000 nM T73725 CV63UL 67240318 IC50 > 10000 nM T73725 C7GRV2 68755406 IC50 > 10000 nM T73725 C5DGR9 69036886 IC50 = 1012 nM T73725 C21JAS 76853169 IC50 = 1600 nM T73725 CU04XY 77105624 IC50 = 2300 nM T73725 CTIA65 77105820 IC50 = 2800 nM T73725 CKB1P9 77106023 IC50 = 44 nM T73725 CXYW85 77106025 IC50 = 610 nM T73725 C2UDS0 77106026 IC50 = 4000 nM T73725 C97SJD 77106027 IC50 = 3500 nM T73725 CFQ10R 77106028 IC50 = 110 nM T73725 CO14DP 77106030 IC50 = 1100 nM T73725 C9G3PA 77106234 IC50 = 3500 nM T73725 CPD27I 77106235 IC50 = 610 nM T73725 CLOR37 77106236 IC50 = 4600 nM T73725 C2GLD8 77106237 IC50 = 400 nM T73725 C0GYK1 86765296 IC50 = 680 nM T73725 C1HW4B 89735655 IC50 = 110 nM T73725 C2LWZ1 129318964 IC50 = 31 nM T73725 C4Z5MQ 131839619 IC50 = 5 nM T73725 C4QM9O 134397095 IC50 = 34 nM T73725 CQ1K2W 134397387 IC50 = 6 nM T73725 CR08AO 134397388 IC50 = 7 nM T73725 CIN73J 134397390 IC50 = 14 nM T73725 C6I1YX 134397391 IC50 = 163 nM T73725 CQ9D1Z 134397392 IC50 = 17 nM T73725 CUX8N5 134397449 IC50 = 26 nM T73725 CDC39N 134397450 IC50 = 120 nM T73725 C8RN6W 134397451 IC50 = 16 nM T73725 CE1HY2 134397452 IC50 = 26 nM T73725 CIR51J 134397453 IC50 = 11 nM T73725 C72KFM 134397463 IC50 = 28 nM T73725 CT16YX 134397502 IC50 = 26 nM T73725 CI45HZ 134397798 IC50 = 92 nM T73725 CI1E8V 137634241 IC50 > 10000 nM T73725 CDA2N6 137644922 IC50 = 5.3 nM T73725 CZ9BN4 138320062 IC50 = 0.261 nM T73725 C5J2WV 138728749 IC50 = 39 nM T73725 CVU63L 139582016 IC50 = 360 nM T73725 C8PH9S 139582017 IC50 = 1400 nM T73725 C6VB3O 145925651 IC50 >= 5000 nM T73725 CX05ZN 145979845 IC50 = 175 nM T73725 CO1S8D 145986658 IC50 = 910 nM T73725 C2MD1Q 155513187 IC50 > 10000 nM T73725 D00ERW 44444843 Ki > 8753 nM T73725 D06CXU 46926513 IC50 = 23 nM T73725 D0D2FC 2794188 IC50 = 111 nM T73725 D0U3NI 53246941 IC50 = 112 nM T73725 D0UI7U 46926514 IC50 = 231 nM T49526 D00BUR 216327 IC50 > 1000 nM T49526 D02AIN 122678117 IC50 > 33000 nM T49526 D0HZ2E 5311271 Ki = 1060 nM T49526 D0K9IF 71666749 IC50 > 30000 nM T49526 C2KDX3 2464255 EC50 = 1470 nM T49526 CKR9Z3 2464257 EC50 > 30000 nM T49526 CRQ37A 4880560 EC50 = 1690 nM T49526 C8T6YH 8762554 EC50 > 30000 nM T49526 CZM2H8 8881840 EC50 > 30000 nM T49526 CS6FN7 9883254 IC50 = 2600 nM T49526 CD34SB 15982534 IC50 = 35000 nM T49526 CU61HC 16827304 EC50 = 2860 nM T49526 CG26CZ 16862803 EC50 > 30000 nM T49526 C7S9NE 25923464 EC50 > 30000 nM T49526 CI1G2C 26873419 IC50 = 2920 nM T49526 C9L4KT 46205341 IC50 > 333000 nM T49526 CL41FE 46206000 IC50 > 333000 nM T49526 CBM42K 53347890 EC50 = 1160 nM T49526 C3YO2J 53347892 EC50 > 30000 nM T49526 C8ZU0D 53347894 EC50 = 1000 nM T49526 C3O7HM 53347896 EC50 = 1410 nM T49526 C94DCG 53347898 EC50 = 7970 nM T49526 CJ9N3F 53347900 EC50 = 1360 nM T49526 CGU48Z 53347904 EC50 = 4740 nM T49526 CZF4S8 53347906 EC50 = 1710 nM T49526 C09ZWT 53347908 EC50 > 30000 nM T49526 C96ZSQ 53347910 EC50 > 30000 nM T49526 C83WFR 53347912 EC50 > 30000 nM T49526 CTOU65 53347914 EC50 > 30000 nM T49526 C7VX8I 53347916 EC50 = 1030 nM T49526 CZY27H 53347918 EC50 = 420 nM T49526 CW9G6X 53347920 EC50 = 6130 nM T49526 CV73XM 53347922 EC50 = 8160 nM T49526 CC45FS 53347924 EC50 = 1780 nM T49526 CC4J5Y 53347926 EC50 = 1380 nM T49526 C9OR6S 53347928 EC50 > 30000 nM T49526 CBZ0Y3 53347930 EC50 = 810 nM T49526 CU90QI 53347932 EC50 = 880 nM T49526 CP1YA3 53488269 EC50 > 30000 nM T49526 C9TM8Q 53488271 EC50 > 30000 nM T49526 CXG6U4 53488272 EC50 > 30000 nM T49526 CZYL42 53488273 EC50 > 30000 nM T49526 CB0RG1 53488275 EC50 = 890 nM T49526 C8APK2 53488280 EC50 = 1630 nM T49526 C4XKH1 53488282 EC50 > 30000 nM T49526 C9BG8K 53488283 EC50 > 30000 nM T49526 CTDY79 53488284 EC50 = 780 nM T49526 CT6UK4 54765372 EC50 = 4380 nM T49526 CXD82U 54765373 EC50 > 30000 nM T49526 CZD5L7 54765374 EC50 > 30000 nM T49526 C72OFG 54765375 EC50 > 30000 nM T49526 C1JMD5 54765376 EC50 = 12900 nM T49526 CU6IC4 54765377 EC50 = 600 nM T49526 C6C5QV 54765378 EC50 > 30000 nM T49526 CA1I6V 54765379 EC50 > 30000 nM T49526 CK8X1W 54765381 EC50 > 30000 nM T49526 CDK50N 54765382 EC50 = 730 nM T49526 C6QKF9 54765445 EC50 > 30000 nM T49526 CAW2J3 54765446 EC50 = 700 nM T49526 C9VH8O 54765447 EC50 = 2590 nM T49526 CYBF21 54765449 EC50 > 30000 nM T49526 C9B2HV 54765450 EC50 > 30000 nM T49526 CKXT78 54765451 EC50 > 30000 nM T49526 C97QTU 54765453 EC50 > 30000 nM T49526 C36HEY 56947221 EC50 = 27400 nM T49526 C2XWQ6 56947223 EC50 = 1320 nM T49526 CLT4Z1 56947228 EC50 > 30000 nM T49526 C5LUY8 56947229 EC50 > 30000 nM T49526 CPR1W3 56947230 EC50 > 30000 nM T49526 CJA45K 56947232 EC50 > 30000 nM T49526 C2POB1 56947233 EC50 > 30000 nM T49526 C1YK2E 122678192 IC50 > 33000 nM T49526 CJH2V9 137637559 IC50 = 2640 nM T49526 C2KX3V 137661020 IC50 > 3000 nM T49526 CKZT21 155559364 IC50 > 33000 nM T49526 D08ATZ 51351551 EC50 = 49290 nM T49526 D0W2FU 53347902 EC50 = 260 nM T12837 CWU8N7 67338 IC50 = 3000 nM T12837 C0O3TQ 126437 IC50 > 400000 nM T12837 C5N0PM 295976 IC50 = 3100 nM T12837 CWF94O 428849 IC50 = 890 nM T12837 CJ2CX8 582689 IC50 > 65000 nM T12837 CQEF34 1002773 IC50 > 100000 nM T12837 C8G4OE 1192043 IC50 > 100000 nM T12837 CV6LA5 2297580 IC50 = 16600 nM T12837 C89ATQ 2779831 IC50 = 1000 nM T12837 CN0F5E 3014812 IC50 = 7500 nM T12837 C8TOU9 3496505 IC50 > 20000 nM T12837 CH9K1U 5351747 IC50 = 400000 nM T12837 CNK84Q 7128991 IC50 = 105000 nM T12837 CEKH37 10979651 IC50 > 400000 nM T12837 CJ6E7G 11087601 IC50 = 20500 nM T12837 C1ZR6H 11848210 IC50 = 1.2 nM T12837 C4QAH6 15342414 IC50 = 1637 nM T12837 C0M7WQ 22390870 IC50 = 98 nM T12837 CJQ86Y 24827559 IC50 = 8600 nM T12837 CJ4IC6 24962989 IC50 = 80 nM T12837 CA7K9P 43167849 IC50 = 1220 nM T12837 CCLQ46 43187900 IC50 = 5310 nM T12837 C0Y9FH 43199381 IC50 = 200 nM T12837 C7F4DG 44574239 IC50 = 60 nM T12837 CPS2T8 44574240 IC50 = 210 nM T12837 C18PTZ 44574241 IC50 = 310 nM T12837 C4V6OX 44574242 IC50 = 1540 nM T12837 CYZ4G1 44574264 IC50 = 50 nM T12837 CJG7H1 44574265 IC50 = 160 nM T12837 C9KMX6 44574266 IC50 = 50 nM T12837 C9WB3L 44574306 IC50 = 50 nM T12837 CL24UR 44574307 IC50 = 130 nM T12837 C6NE3R 44574308 IC50 = 2200 nM T12837 CQI27O 44574309 IC50 = 400 nM T12837 CJ6L4K 44574374 IC50 = 360 nM T12837 C1RIT4 44574375 IC50 = 2100 nM T12837 C98OJN 44574376 IC50 > 10000 nM T12837 CHI9F3 44574377 IC50 > 10000 nM T12837 C12DMU 44578429 IC50 = 10600 nM T12837 C5GCR8 44578430 IC50 = 29800 nM T12837 C04YVX 44578431 IC50 = 7700 nM T12837 C0WB8T 44578432 IC50 = 230 nM T12837 C8AIP0 44578462 IC50 = 1420 nM T12837 C5N3CJ 44578463 IC50 = 16900 nM T12837 CX4YR8 44578464 IC50 = 160 nM T12837 C3P2UH 44578465 IC50 = 20100 nM T12837 CI0NP8 44578466 IC50 > 30000 nM T12837 CNU74O 44578467 IC50 > 30000 nM T12837 C7ZQW8 44578468 IC50 > 30000 nM T12837 CRSC45 44578469 IC50 = 1320 nM T12837 CI2O0T 44578470 IC50 = 3400 nM T12837 CX95VH 44578502 IC50 = 7100 nM T12837 C92YUQ 44578503 IC50 = 180 nM T12837 CQO7X6 44578504 IC50 = 1100 nM T12837 CZ1F4S 44578505 IC50 = 4300 nM T12837 CZE1J7 44578539 IC50 = 1800 nM T12837 C8GZB2 44578540 IC50 > 50000 nM T12837 CJTR68 44578541 IC50 > 50000 nM T12837 CMQ5N2 44578542 IC50 = 600 nM T12837 CQA74O 45487305 IC50 > 30 nM T12837 CJZ41I 45487306 IC50 > 30 nM T12837 CABH45 45487323 IC50 = 0.12 nM T12837 CD4OH6 45487347 IC50 = 0.26 nM T12837 CEA04X 45487348 IC50 = 2.9 nM T12837 CLP03M 45487354 IC50 = 0.7 nM T12837 CYJ42A 45487360 IC50 = 0.84 nM T12837 CXD72H 45487361 IC50 = 0.41 nM T12837 CD36FG 45487378 IC50 = 17 nM T12837 CA9GE3 45487379 IC50 = 4.6 nM T12837 CWHP79 46867603 IC50 = 30 nM T12837 C70ZYQ 46997620 IC50 = 11100 nM T12837 CUA83Y 50937454 IC50 = 27 nM T12837 CN01BZ 53211571 IC50 > 4700 nM T12837 CKAI31 53361222 IC50 = 8100 nM T12837 CV25JZ 53361223 IC50 = 14400 nM T12837 C0C6YK 53363652 IC50 = 10300 nM T12837 CPU86Z 53363653 IC50 = 15200 nM T12837 C63DVR 53363743 IC50 = 11900 nM T12837 COBL07 53363744 IC50 = 12500 nM T12837 C8QFS7 53363745 IC50 = 12200 nM T12837 CEG3P9 53363834 IC50 = 14800 nM T12837 CW4CD0 53363835 IC50 = 16000 nM T12837 C02ORV 53377508 Ki > 20000 nM T12837 CYM2T4 53868701 IC50 = 32 nM T12837 CPL71I 54596764 IC50 = 116000 nM T12837 C0YR1M 55070650 IC50 > 10000 nM T12837 C72GHW 56642706 IC50 > 100000 nM T12837 CS6Q7R 56642708 IC50 > 100000 nM T12837 CC2O7Y 56746673 IC50 = 13300 nM T12837 C3FUP7 56753262 IC50 = 1900 nM T12837 C7VQ5F 56759179 IC50 > 30000 nM T12837 CN7V5L 56759225 IC50 > 40000 nM T12837 CRI9T6 56759592 IC50 = 600 nM T12837 CJBY70 56951879 Ki > 50000 nM T12837 CD6V9F 58730746 IC50 = 6250 nM T12837 C04KFR 60150359 IC50 = 3000 nM T12837 CQ60CT 62206064 IC50 = 2460 nM T12837 C7RJD3 63155127 IC50 = 3190 nM T12837 CNR16Q 63189585 IC50 > 10000 nM T12837 CQ27KW 64381918 IC50 = 8340 nM T12837 CER5F1 67466175 IC50 > 100000 nM T12837 CO6L5Z 67739618 IC50 = 80 nM T12837 C5QE6A 67988955 IC50 > 50000 nM T12837 C8JTS3 70676140 Ki > 100000 nM T12837 CZL47S 70676141 Ki > 100000 nM T12837 C8KC6O 70676142 Ki > 100000 nM T12837 CAFU69 70686225 IC50 = 100000 nM T12837 CM53OA 72918546 IC50 > 50000 nM T12837 CUP4Q6 76328021 Ki > 50000 nM T12837 CX7V5M 76328022 Ki > 50000 nM T12837 C5P2BM 76331683 Ki > 50000 nM T12837 C8KEM3 91645136 IC50 = 360 nM T12837 C73LWN 92136227 IC50 = 4 nM T12837 CWG18C 118731739 IC50 = 7230 nM T12837 CI1AE0 118731742 IC50 = 5800 nM T12837 C6Y8BM 118731746 IC50 = 21500 nM T12837 CIOL82 122195095 IC50 = 10000 nM T12837 C6KV9H 124081151 IC50 = 50 nM T12837 CP94YL 127031964 IC50 = 27 nM T12837 C9KJ2Q 134130626 IC50 = 149 nM T12837 CV95CT 134131930 IC50 = 3680 nM T12837 CIV51H 134132630 IC50 = 177 nM T12837 C3W8IS 134132824 IC50 = 16 nM T12837 CJ8H7W 134134884 IC50 = 14 nM T12837 CFVI01 134135475 IC50 = 1540 nM T12837 CIY91H 134135786 IC50 = 85 nM T12837 CBJ1S8 134137030 IC50 = 108 nM T12837 CT5I6V 134137361 IC50 = 62 nM T12837 C13UJH 134137680 IC50 = 28 nM T12837 C0C4AO 134138246 IC50 = 53 nM T12837 C4AFS3 134140748 IC50 = 35 nM T12837 CF57RU 134140884 IC50 = 120 nM T12837 CP59XG 134141266 IC50 = 19 nM T12837 C38BUI 134141657 IC50 = 616 nM T12837 CG8PM2 134142051 IC50 = 23 nM T12837 CKGL61 134142579 IC50 = 33 nM T12837 CPS6D3 134144201 IC50 = 18 nM T12837 C2GC5B 134144476 IC50 = 41 nM T12837 C67DQZ 134144962 IC50 = 15 nM T12837 CSY51N 134146326 IC50 = 18 nM T12837 CRY2Z5 134146985 IC50 = 41 nM T12837 C8L6ZH 134148531 IC50 = 15 nM T12837 CEAV71 134149335 IC50 = 42 nM T12837 C5U6TX 134151277 IC50 = 103 nM T12837 C0PIN9 134153830 IC50 = 1070 nM T12837 CMHQ35 134153978 IC50 = 27 nM T12837 C8UX3L 134154872 IC50 = 231 nM T12837 C2OR9A 134155520 IC50 = 17 nM T12837 C54FUD 134155964 IC50 = 28 nM T12837 CXM26R 134156697 IC50 = 22 nM T12837 CF3GA7 134157655 IC50 = 17 nM T12837 CDXJ59 136180348 IC50 = 2600 nM T12837 C93QGH 137633458 IC50 = 69 nM T12837 C4LK1X 137635057 IC50 = 94 nM T12837 C1PMC9 137636992 IC50 = 94 nM T12837 CJ4Q8Z 137638223 IC50 = 223 nM T12837 C13YKS 137638371 IC50 = 130 nM T12837 C8FZG6 137642809 IC50 = 90 nM T12837 C16DLH 137647272 IC50 = 302 nM T12837 C51RHP 137647665 IC50 = 67 nM T12837 C1O5PE 137652170 IC50 = 342 nM T12837 CCO6Z7 137654377 IC50 = 330 nM T12837 CRT8Q3 137655207 IC50 = 63 nM T12837 CK7BA8 137656269 IC50 = 157 nM T12837 C9Z6GL 137659934 IC50 = 144 nM T12837 CB9FM8 137661596 IC50 = 50 nM T12837 CDPN65 137661881 IC50 = 471 nM T12837 CR5D4S 138753329 IC50 = 480 nM T12837 C51ILK 138753330 IC50 = 2000 nM T12837 CE58DF 153041236 IC50 > 100000 nM T12837 CC50SM 155511980 IC50 = 130 nM T12837 CTM72I 155513465 IC50 = 240 nM T12837 C78OZR 155516239 IC50 = 4260 nM T12837 CJQH26 155516447 IC50 = 465 nM T12837 CU04SF 155519144 IC50 = 279 nM T12837 CH5J9U 155520755 IC50 = 6120 nM T12837 C6CY0R 155523571 IC50 = 120 nM T12837 C2LRU6 155523638 IC50 = 1990 nM T12837 C4JEC2 155526486 IC50 = 220 nM T12837 CKNF47 155527838 IC50 = 2310 nM T12837 CTHM63 155528468 IC50 = 11600 nM T12837 C5BUY9 155529011 IC50 = 101 nM T12837 C7C8HI 155529624 IC50 = 21 nM T12837 CBU23P 155531094 IC50 = 2070 nM T12837 C7U9IT 155534335 IC50 = 410 nM T12837 CYMG91 155534360 IC50 = 270 nM T12837 CY8O0Q 155535049 IC50 = 475 nM T12837 CZRU49 155535884 IC50 = 1700 nM T12837 C70HAX 155536607 IC50 = 4480 nM T12837 C0RY3I 155538329 IC50 = 2310 nM T12837 C67JQV 155538900 IC50 > 200000 nM T12837 CO03YQ 155541365 IC50 = 270 nM T12837 CY2W3F 155541904 IC50 = 600 nM T12837 C8LZ6X 155542642 IC50 = 1950 nM T12837 C4UT5G 155542694 IC50 = 785 nM T12837 CYO70M 155543486 IC50 = 3820 nM T12837 CNLE45 155543945 IC50 = 1180 nM T12837 CPXC10 155546110 IC50 = 305 nM T12837 C08EQC 155546573 IC50 = 43 nM T12837 CQ9A0Z 155547391 IC50 = 3490 nM T12837 CHB87K 155547731 IC50 = 658 nM T12837 CKUV39 155549017 IC50 = 37 nM T12837 CM4C9U 155549658 IC50 = 343 nM T12837 C79QNS 155549883 IC50 = 254 nM T12837 CJ8ZI6 155549992 IC50 = 51000 nM T12837 CHPG47 155551515 IC50 = 2050 nM T12837 CVN57A 155552644 IC50 = 5220 nM T12837 C3Q7YP 155558960 IC50 = 900 nM T12837 C3PMG9 155559000 IC50 = 31 nM T12837 CEI8R4 155559940 IC50 = 7980 nM T12837 CU06YI 155562437 IC50 = 165 nM T12837 C8LKQ6 155564730 IC50 = 2610 nM T12837 C81NJP 155565393 IC50 = 772 nM T12837 CTCM91 155566361 IC50 = 530 nM T12837 CF4ZI2 155567058 IC50 = 228 nM T12837 CW56PR 155567067 IC50 = 2130 nM T12837 CVJ62X 155568483 IC50 = 2110 nM T12837 C47PWI 46905055 IC50 > 50000 nM T12837 D02TVQ 71268957 IC50 = 128000 nM T12837 D09CLP 439155 Ki = 400 nM T12837 D0A1CM 5281855 IC50 = 25000 nM T12837 D0BU8W 44219611 IC50 = 0.04 nM T12837 D0Q3FY 44622850 IC50 = 0.07 nM T72458 D0G2XE 6918468 IC50 = 400 nM T72458 D0H7AR 70684954 Ki = 26000 nM T72458 D0LI1C 44469321 IC50 > 30000 nM T72458 D0X9PF 9941379 EC50 = 0.2 nM T72458 CA3ZU6 489667 IC50 = 612 nM T72458 CZN6S9 743974 EC50 > 31622.78 nM T72458 CL04VQ 910537 Ki > 1000000 nM T72458 C0DA9X 2163781 Ki = 161000 nM T72458 CK4YT2 2817655 Ki > 1000000 nM T72458 CB9A2M 2852098 Ki = 118000 nM T72458 C8EPT1 6918707 EC50 = 4 nM T72458 CWZ1O2 6918780 EC50 = 0.44 nM T72458 CY60AZ 6918813 EC50 = 6 nM T72458 C2BQE1 6918814 Ki = 1.8 nM T72458 CK83QR 6918844 Ki = 3.2 nM T72458 C14CGB 6918847 Ki = 6.3 nM T72458 CLV3C7 6918849 IC50 = 0.77 nM T72458 C5U7CS 6918850 Ki = 2.8 nM T72458 C0Q5JL 6918851 IC50 = 8 nM T72458 CRG04O 6918857 Ki = 20 nM T72458 COS6C1 9808720 EC50 = 11 nM T72458 CM02VS 9808801 EC50 = 13 nM T72458 C8IM6O 9851816 Ki = 12.9 nM T72458 CVM3K1 9852314 Ki = 600 nM T72458 CKCF18 9867330 EC50 = 16 nM T72458 CM3Y5H 9893728 IC50 = 9157 nM T72458 CZ5E2C 9915636 Ki = 20.5 nM T72458 CCL2T8 9915813 EC50 = 2600 nM T72458 CFG0W2 9917301 IC50 = 118 nM T72458 CNF37L 9919056 EC50 = 2 nM T72458 C15DES 9924916 Ki = 140000 nM T72458 C7V8AE 9946241 Ki = 42000 nM T72458 CX5CU3 9958649 Ki = 590 nM T72458 C97MRJ 9960253 EC50 = 16 nM T72458 CMU31X 9968756 Ki = 27000 nM T72458 C5F3QU 9969456 Ki = 6400 nM T72458 C5U0JO 9977350 Ki = 180 nM T72458 CG58RO 9983075 Ki = 190 nM T72458 CR6TX4 10004020 IC50 = 52 nM T72458 CC48YG 10008561 EC50 = 6700 nM T72458 CLXA58 10025669 Ki = 25118.86 nM T72458 CRP4X1 10030530 Ki = 6 nM T72458 CL2PE9 10031074 Ki = 2500 nM T72458 C8KI2R 10033237 Ki = 160 nM T72458 CGJ72R 10049407 Ki = 770 nM T72458 C9YQS5 10050686 Ki = 89 nM T72458 CMGB68 10053261 Ki = 6300 nM T72458 CAG52F 10072440 Ki = 920 nM T72458 CSH3Y2 10075878 IC50 = 530 nM T72458 CZ78WX 10077258 EC50 = 13 nM T72458 C7T2XW 10077483 Ki = 4100 nM T72458 CUR4Y1 10077594 Ki = 57 nM T72458 C8MCA1 10077773 Ki = 1.95 nM T72458 C7PV4C 10098133 EC50 = 240 nM T72458 CP5H2J 10098568 IC50 = 260 nM T72458 CW4E8K 10101361 EC50 = 2.17 nM T72458 CSQ60B 10108894 Ki = 16000 nM T72458 C6LVA2 10109225 Ki = 5000 nM T72458 C0DP3Z 10117829 IC50 = 871 nM T72458 C8AQP5 10119206 EC50 = 40 nM T72458 CG1K8Y 10122170 EC50 < 0.1 nM T72458 CFX6U7 10123761 EC50 = 33 nM T72458 C6Y3KL 10128451 IC50 = 16 nM T72458 CF81WV 10132207 Ki = 66000 nM T72458 C0PVS9 10134057 Ki = 6200 nM T72458 CC0ZT7 10137615 Ki = 16000 nM T72458 C86FWN 10141778 IC50 = 16 nM T72458 C2AF5L 10146090 IC50 = 12 nM T72458 CO69QN 10146211 EC50 = 0.58 nM T72458 C51LKY 10146483 EC50 = 65 nM T72458 C03AKT 10155513 Ki = 67000 nM T72458 CPRS08 10157774 Ki = 13000 nM T72458 CXF16O 10158674 Ki = 62000 nM T72458 C97IHD 10159196 Ki = 12000 nM T72458 C1XJM3 10165866 IC50 = 12 nM T72458 CX7WV9 10168556 EC50 = 120 nM T72458 CTD14O 10169912 EC50 = 9 nM T72458 CAB06U 10177247 Ki = 161000 nM T72458 COJ1M5 10178845 Ki = 6800 nM T72458 CV2QX0 10180932 Ki = 12000 nM T72458 C78FGS 10188529 IC50 = 28 nM T72458 C1HMR6 10200110 Ki = 111000 nM T72458 CFZ5I6 10210964 IC50 = 1.9 nM T72458 C8PA3J 10211466 Ki = 73.7 nM T72458 C1VCQ8 10213106 EC50 = 13 nM T72458 CWJ5I0 10225762 Ki = 25000 nM T72458 CH67VW 10230144 IC50 = 30 nM T72458 CF8SA2 10232394 IC50 = 11 nM T72458 CTO7I8 10232787 Ki = 7.3 nM T72458 CFH82K 10239507 IC50 = 11.2 nM T72458 C1OYR8 10255546 Ki = 2600 nM T72458 CSNY06 10257242 EC50 = 25 nM T72458 C6Y1ER 10257541 Ki = 1 nM T72458 C2AL7S 10260053 Ki = 630 nM T72458 CEC2M0 10269187 Ki = 74000 nM T72458 C6T2MU 10270570 Ki = 11000 nM T72458 CX29KB 10282847 IC50 = 1.1 nM T72458 C4SCW2 10283036 Ki = 5.8 nM T72458 CBL5E0 10283067 Ki = 6.4 nM T72458 C01QVJ 10291369 Ki = 26000 nM T72458 CSDX25 10291370 Ki = 7400 nM T72458 CX97KY 10292084 Ki = 33000 nM T72458 C7WDA8 10292876 Ki = 7000 nM T72458 CU17RB 10293285 Ki = 16000 nM T72458 CV3ZJ5 10304463 Ki = 95.6 nM T72458 CU13DH 10304547 IC50 = 0.37 nM T72458 C1E3PC 10304776 IC50 = 1.1 nM T72458 CC0N9A 10304794 Ki = 5.3 nM T72458 CU0CH8 10324857 Ki = 4.3 nM T72458 CE4OK9 10325306 Ki = 0.83 nM T72458 CT9AR6 10325955 EC50 = 14 nM T72458 CO40LC 10348630 EC50 = 227 nM T72458 CSH89D 10369375 Ki = 3.2 nM T72458 C84RZU 10373417 EC50 = 2 nM T72458 C1N3MA 10392968 IC50 = 1900 nM T72458 CJN2I7 10411266 Ki = 340 nM T72458 CNK7M3 10414731 Ki = 80 nM T72458 CPL02I 10463896 EC50 = 6.08 nM T72458 C1GJ2S 10481801 IC50 = 152 nM T72458 CS2EQ0 10481883 Ki = 11 nM T72458 CTEB92 10483153 EC50 = 18 nM T72458 C3NWO8 10484741 EC50 = 59 nM T72458 CICJ50 10864263 IC50 = 469 nM T72458 CBPX36 10864861 EC50 = 8.7 nM T72458 C5SK0I 10874535 IC50 = 597 nM T72458 CM5GF3 10886436 IC50 = 3050 nM T72458 CGIC31 10918643 IC50 = 2081 nM T72458 C52NZB 10928744 IC50 = 193 nM T72458 CP6WR3 10951027 IC50 = 266 nM T72458 CN9D6B 10952071 IC50 = 127 nM T72458 COE81Y 10973172 IC50 = 150 nM T72458 CJKA90 10996121 EC50 = 297 nM T72458 CY3TJ1 10996232 EC50 = 32 nM T72458 CQJF15 11016325 IC50 = 3226 nM T72458 CAL9N7 11017471 Ki = 1.2 nM T72458 C7IJV5 11038873 EC50 = 630 nM T72458 CA2X6S 11050211 IC50 = 238 nM T72458 CHOS10 11061068 IC50 = 0.3 nM T72458 CNP78D 11092487 IC50 = 249 nM T72458 C5H7IP 11092574 IC50 = 364 nM T72458 CO2U6S 11156852 EC50 = 274 nM T72458 C4V9OW 11157584 Ki = 14 nM T72458 CF6T8V 11158829 EC50 = 1995.26 nM T72458 C81JOX 11170774 EC50 = 29 nM T72458 CG64NJ 11179914 EC50 = 490 nM T72458 C3V7DK 11180881 Ki = 15 nM T72458 CHC51K 11181804 Ki = 10.8 nM T72458 CDLG18 11205265 EC50 = 1995.26 nM T72458 C9WTR4 11205266 EC50 = 63.1 nM T72458 CDMB38 11205293 EC50 = 794.33 nM T72458 CLJ83I 11205294 EC50 = 1995.26 nM T72458 C0F8CB 11214733 EC50 = 145 nM T72458 CUC85X 11215553 EC50 = 3.2 nM T72458 CD5SG6 11215758 Ki = 4.8 nM T72458 CF7VQ4 11226756 EC50 = 7 nM T72458 CWLJ34 11237444 Ki = 1300 nM T72458 CR1Q2X 11237928 EC50 = 150 nM T72458 C30NWM 11238126 EC50 = 40 nM T72458 C1T3VM 11249545 Ki = 840 nM T72458 CD5YZ2 11249788 EC50 = 44 nM T72458 C6FBD3 11251566 EC50 = 158.49 nM T72458 C6ETW3 11251567 EC50 = 1258.93 nM T72458 C9LOV4 11251591 EC50 = 251.19 nM T72458 CMI4E5 11251592 EC50 = 79.43 nM T72458 CE2P7Y 11261324 EC50 = 210 nM T72458 CF58GC 11262020 EC50 = 140 nM T72458 C0D1PE 11263072 EC50 = 2.512 nM T72458 CMS1L8 11272336 EC50 = 200 nM T72458 CP9S6F 11273288 EC50 = 2 nM T72458 C07VJD 11274575 IC50 = 158.49 nM T72458 CS2U3A 11286048 IC50 = 1995.26 nM T72458 CS57OX 11295536 EC50 = 71 nM T72458 CQ47NA 11295737 EC50 = 110 nM T72458 CJ7OT2 11296600 EC50 = 3.8 nM T72458 C2PU1F 11296732 Ki = 44 nM T72458 CYH1I3 11297620 EC50 < 0.01 nM T72458 C9XBQ7 11308054 Ki = 29 nM T72458 CYK4F0 11308184 Ki = 77 nM T72458 C97ICV 11309021 IC50 = 794.33 nM T72458 CVE6D9 11309022 EC50 = 794.33 nM T72458 CO0C7R 11330869 Ki = 27 nM T72458 CYUL15 11330992 EC50 = 8 nM T72458 CS7K4R 11341045 Ki = 650 nM T72458 CU6Y1Z 11341046 Ki = 1500 nM T72458 C3RI8D 11341811 EC50 = 34 nM T72458 C4OEC6 11353522 EC50 = 93 nM T72458 CHWO84 11353851 EC50 = 400 nM T72458 CAL3F9 11364326 Ki = 580 nM T72458 C41ZBP 11364343 EC50 = 1300 nM T72458 CYVD37 11364802 EC50 = 44 nM T72458 CEX40J 11366515 EC50 = 630.96 nM T72458 CZ6RU2 11375529 EC50 = 360 nM T72458 C5D1TY 11375764 Ki = 840 nM T72458 C6SN4C 11378005 EC50 = 1258.93 nM T72458 CV7BU3 11378006 EC50 = 1995.26 nM T72458 CR8B4G 11378033 EC50 = 316.23 nM T72458 CUPS87 11387898 EC50 = 150 nM T72458 CMF98X 11398483 Ki = 37 nM T72458 CQ1ZL6 11411962 IC50 = 398.11 nM T72458 CQ7WS5 11421919 Ki = 24 nM T72458 CUTZ31 11445925 EC50 = 398.11 nM T72458 C0GFV8 11456260 EC50 = 48 nM T72458 C3FML2 11468019 Ki = 69.5 nM T72458 C2DNI1 11468666 EC50 = 158.49 nM T72458 C8LN5W 11477853 Ki = 1400 nM T72458 CG5D6C 11480040 IC50 = 3981.07 nM T72458 CPT4K8 11490215 EC50 = 98 nM T72458 CVR0T4 11490658 Ki = 6.3 nM T72458 CY8AJ5 11512024 EC50 = 281.84 nM T72458 CKE15O 11555886 EC50 = 17.9 nM T72458 CF7NS4 11571540 EC50 = 1 nM T72458 CA5GQ7 11592389 EC50 = 151.36 nM T72458 CL87NX 11593230 EC50 = 1 nM T72458 C24UQH 11599302 EC50 = 44.67 nM T72458 CDP3W4 11607111 EC50 = 40 nM T72458 CR0N5C 11613526 EC50 = 707.95 nM T72458 C7F9XQ 11613741 EC50 = 354.81 nM T72458 COLB48 11627577 EC50 = 3235.94 nM T72458 CRE2X6 11635051 EC50 = 537.03 nM T72458 C7JU6O 11635265 EC50 = 177.83 nM T72458 CM2A6K 11636019 Ki = 16 nM T72458 CPM61U 11685018 EC50 = 323.59 nM T72458 C3XN4O 11692334 EC50 = 436.52 nM T72458 C6WAM2 11706338 EC50 = 1000 nM T72458 CWZX95 11730771 IC50 = 1500 nM T72458 C6GMS7 11732821 IC50 > 5000 nM T72458 C3NWA7 11733360 IC50 = 336 nM T72458 C5AZ2R 11753667 EC50 = 21 nM T72458 CIHY70 11753668 EC50 = 44 nM T72458 CH7TQ6 11753695 EC50 = 4.6 nM T72458 C63DVB 11756904 Ki = 64 nM T72458 C59XUF 11757528 EC50 = 710 nM T72458 CHI2W5 11761948 IC50 > 10000 nM T72458 CUL54T 11764499 EC50 = 100 nM T72458 C2SHV7 11786860 EC50 = 12 nM T72458 CD9N5B 11787842 EC50 = 501.19 nM T72458 CQ06HS 11787864 EC50 = 316.23 nM T72458 CMJ3K5 11811937 IC50 = 3829 nM T72458 C0OIV9 11813437 EC50 = 840 nM T72458 C7NL4J 11845272 Ki = 10 nM T72458 C4XF1I 11845276 Ki = 137 nM T72458 CT1F9R 11845438 EC50 = 97 nM T72458 CC42HM 11845440 EC50 = 501 nM T72458 CFKN79 11845444 Ki = 2353 nM T72458 C3JV7M 11845450 EC50 = 2.3 nM T72458 C8WJ6E 11845630 EC50 = 252 nM T72458 CI1VU0 11845804 EC50 = 986 nM T72458 C4V9DO 11845813 EC50 = 291 nM T72458 CSZX65 11846669 EC50 = 14 nM T72458 C5HFB2 11846673 Ki = 90 nM T72458 C25KCW 11846844 EC50 = 39 nM T72458 CO3H9V 11847001 EC50 = 9 nM T72458 CECQ63 11847312 EC50 = 292 nM T72458 C91GMR 11851038 EC50 = 1.02 nM T72458 CT4EC3 11966875 IC50 > 10000 nM T72458 CG15NA 15602927 IC50 = 90 nM T72458 C0E4PU 15603023 IC50 = 60 nM T72458 CI9W3G 15953833 IC50 = 1.5 nM T72458 CAT74W 15953838 EC50 = 177 nM T72458 C2BLT4 16007263 EC50 = 1.7 nM T72458 C54MIL 16007264 Ki = 19 nM T72458 C6XS3N 16007285 Ki = 13 nM T72458 CK3T2B 16038121 EC50 = 1113.1 nM T72458 CYW0B8 16038315 Ki = 6.7 nM T72458 CSM3L8 16038316 Ki = 10 nM T72458 C4N0VF 16046215 Ki = 25 nM T72458 CX68DN 16049796 EC50 > 10000 nM T72458 C8UXP9 16126683 EC50 = 29.7 nM T72458 CPTO16 16132144 EC50 = 0.21 nM T72458 C9YZE5 16133802 EC50 = 0.65 nM T72458 CM8QO6 16721030 IC50 = 19.8 nM T72458 CZU6Q0 16725558 EC50 = 214.5 nM T72458 C4NZ3C 16725559 IC50 = 3.3 nM T72458 CR1DM4 16746686 IC50 = 0.84 nM T72458 C7WHL3 16746823 EC50 = 0.11 nM T72458 C25XZF 17880880 Ki > 1000000 nM T72458 CW58XN 22318631 IC50 = 131 nM T72458 C8BY2K 22318635 IC50 = 40.3 nM T72458 CCQ0V9 22318636 IC50 = 22 nM T72458 CG5SO7 22318639 IC50 = 72.3 nM T72458 C8BFU5 22318643 IC50 = 3590 nM T72458 C6MID9 22318657 IC50 = 303 nM T72458 C9QO2V 22318671 IC50 = 263 nM T72458 CZ1GJ8 23634985 Ki = 35 nM T72458 C6UP8O 23634986 Ki = 9.7 nM T72458 C0RM6I 23635105 Ki = 69 nM T72458 CB45UM 23635106 Ki = 6 nM T72458 CFNQ06 23635107 Ki = 2.8 nM T72458 CPE8L0 23635108 Ki = 2.2 nM T72458 CDC19H 23635109 Ki = 0.6 nM T72458 CHU29W 23635235 Ki = 2.8 nM T72458 CWL5K4 23635236 Ki = 5.7 nM T72458 CVFQ41 23635237 Ki = 5.9 nM T72458 CBW09O 23653113 Ki = 16000 nM T72458 C8KO9M 23661656 Ki = 11 nM T72458 C7DW6E 24180493 EC50 = 4.6 nM T72458 CK2Q5J 24180592 Ki = 3.4 nM T72458 C0QI2D 24180593 Ki = 0.9 nM T72458 C7SMW5 24180646 Ki = 0.9 nM T72458 CC4FM5 24740310 Ki = 890 nM T72458 CGY27Z 24740311 Ki = 260 nM T72458 CE6D9F 24740312 Ki = 6 nM T72458 CU19BT 24740419 Ki = 2.5 nM T72458 C2K1EL 24740535 Ki = 3.2 nM T72458 CTC05L 24740653 Ki = 3.7 nM T72458 CD90WZ 24740655 Ki = 0.59 nM T72458 CUPD43 24741624 Ki = 14 nM T72458 C2S3RO 24741625 Ki = 9.7 nM T72458 C52ZAS 24741961 Ki = 36 nM T72458 CT4I7Z 24741964 Ki = 39 nM T72458 CB47WZ 24764421 IC50 = 19.7 nM T72458 C5TA3W 24774358 IC50 = 160 nM T72458 CO4JK2 24774437 IC50 > 10000 nM T72458 CMB27G 24774521 IC50 = 520 nM T72458 C2TAK6 24774601 IC50 > 1000 nM T72458 C59NIQ 24848934 EC50 = 1.8 nM T72458 C2A1SX 24848995 EC50 = 80 nM T72458 C1EN7W 24857886 IC50 = 7.8 nM T72458 CB9M3F 24873537 Ki = 11 nM T72458 CS0L2N 24882666 Ki = 4200 nM T72458 CP2X4S 24886259 Ki = 6.8 nM T72458 CJ96SC 24886260 Ki = 12.7 nM T72458 CI37TV 24886498 Ki = 27.3 nM T72458 C1M8NX 24886499 Ki = 15.6 nM T72458 CU38LE 24886501 Ki = 75.8 nM T72458 C6IV8J 24886734 Ki = 31.4 nM T72458 C0YV3J 24886735 Ki = 70 nM T72458 CPQ74G 25022598 Ki = 1.1 nM T72458 CG9AV5 25058412 Ki = 8.1 nM T72458 CV07PW 25108215 EC50 = 0.28 nM T72458 CJ5HN6 25128748 EC50 = 37 nM T72458 C3WE0T 25128749 EC50 = 3 nM T72458 CP5TN2 25128751 Ki = 36 nM T72458 CUTA14 25129105 Ki = 6 nM T72458 CPL49Z 25129107 EC50 = 1.2 nM T72458 C4N5DH 25129108 EC50 = 9 nM T72458 CDC2Q6 25129109 EC50 = 1.7 nM T72458 CVSO97 25129453 EC50 = 0.8 nM T72458 CE79VX 25131477 EC50 = 391 nM T72458 C1B7KF 25131478 EC50 = 0.9 nM T72458 CIJ6P4 25132524 EC50 = 31 nM T72458 CY42MT 25132525 EC50 = 83 nM T72458 C9QG3J 25132526 EC50 = 8 nM T72458 CL3JV6 25132864 EC50 = 5 nM T72458 C57QZT 25132866 Ki = 4 nM T72458 CR6YZ2 25132867 EC50 = 25 nM T72458 C8AO5Y 25133207 Ki = 26 nM T72458 C3VGX6 25133208 EC50 = 10 nM T72458 C3KRA8 25133209 EC50 = 2.7 nM T72458 C9U6CQ 25133210 EC50 = 0.9 nM T72458 C74ACT 25133556 EC50 = 1.3 nM T72458 CW7O1N 25133903 EC50 = 167 nM T72458 CG3R0Y 25133907 EC50 = 28 nM T72458 C4SH1P 25211670 Ki = 9.6 nM T72458 CE01RM 25217223 Ki = 416.87 nM T72458 C8O1PH 25217225 Ki = 45 nM T72458 C4HK6C 42630327 EC50 < 0.03162 nM T72458 CU4S6X 44157099 IC50 = 2.5 nM T72458 CBG73U 44158097 EC50 = 43 nM T72458 CIOF26 44158168 IC50 = 0.6 nM T72458 C53LJK 44158169 IC50 = 5.7 nM T72458 CF7X1N 44158255 EC50 = 250 nM T72458 C9UD8I 44158336 EC50 = 200 nM T72458 CF6PT4 44158337 IC50 = 1.5 nM T72458 CHKI60 44265225 Ki > 1000000 nM T72458 CXN2R4 44265309 Ki = 94000 nM T72458 C3EJ1R 44265312 Ki = 161000 nM T72458 CWPT03 44265315 Ki = 24000 nM T72458 CJ1M6N 44265347 Ki = 44000 nM T72458 CEQ6K7 44265351 Ki = 89000 nM T72458 CSL48C 44265374 Ki = 2000 nM T72458 C97AIK 44265472 Ki = 107000 nM T72458 C6DZ4W 44265473 Ki = 8800 nM T72458 CLE96R 44265479 Ki = 68000 nM T72458 CV8GX6 44265487 Ki = 56000 nM T72458 C2CPG9 44265489 Ki = 104000 nM T72458 CLP5G3 44265496 Ki = 2100 nM T72458 C51TPY 44265586 Ki > 1000 nM T72458 CH5WM7 44265588 Ki > 1000 nM T72458 CT89LY 44265589 Ki = 105000 nM T72458 CZS3C7 44265590 Ki = 134000 nM T72458 C3YKG9 44265591 Ki = 56000 nM T72458 C74SBD 44265625 Ki > 1000 nM T72458 CRQ92O 44265626 Ki > 1000 nM T72458 CT2S8I 44265639 Ki = 6800 nM T72458 C18JZD 44265656 Ki = 205000 nM T72458 CZWE24 44265658 Ki = 66000 nM T72458 CD8UC0 44265662 Ki > 1000 nM T72458 C6OU7D 44265665 Ki > 1000 nM T72458 CC28FH 44265672 Ki = 9900 nM T72458 CSK9V6 44265674 Ki > 1000 nM T72458 CS46LN 44265675 Ki > 1000000 nM T72458 C9E0TB 44265681 Ki = 279000 nM T72458 CCGI15 44265707 Ki = 15000 nM T72458 CION54 44265708 Ki > 1000000 nM T72458 C9CM8W 44265711 Ki = 64000 nM T72458 CPUO61 44265713 Ki = 150000 nM T72458 CP1E6X 44265715 Ki = 14000 nM T72458 CRFQ64 44265719 Ki > 1000000 nM T72458 CXUI50 44265722 Ki = 127000 nM T72458 CVEG42 44265727 Ki > 1000 nM T72458 CC4S8V 44265739 Ki > 1000 nM T72458 CG1CH0 44265748 Ki > 1000 nM T72458 C82FPN 44265749 Ki = 139000 nM T72458 C05MIH 44265751 Ki = 30000 nM T72458 CP82FI 44265757 Ki > 1000 nM T72458 CE6A0Z 44265759 Ki > 1000 nM T72458 CPE83Q 44269189 EC50 = 23 nM T72458 CCP5L2 44269214 EC50 = 77 nM T72458 CN5TI2 44269217 EC50 = 2.9 nM T72458 C4M2LJ 44269245 EC50 = 40 nM T72458 C6LD9E 44275119 EC50 = 35 nM T72458 C60GXU 44275121 EC50 = 33 nM T72458 CFIT54 44275175 EC50 = 7 nM T72458 CO7KR8 44275191 EC50 = 37 nM T72458 C72TAL 44275192 EC50 = 15 nM T72458 CA7DX2 44275263 EC50 = 4 nM T72458 CK4E6O 44275264 EC50 = 176 nM T72458 CB4WG5 44275265 EC50 = 10 nM T72458 C3SH7Q 44275312 EC50 = 48 nM T72458 CIA54K 44275371 EC50 = 45 nM T72458 CBS9X6 44275372 EC50 = 7 nM T72458 C5RJ3Z 44275488 EC50 = 6 nM T72458 CBW0I1 44275650 EC50 = 0.9 nM T72458 CO9BJ6 44275654 EC50 = 65 nM T72458 COUM34 44275656 EC50 = 2 nM T72458 CSI8T3 44277299 EC50 = 120 nM T72458 CCGT80 44277300 EC50 = 90 nM T72458 CLG8Y1 44277301 EC50 = 130 nM T72458 C5OHC4 44277696 EC50 = 20 nM T72458 CMU9P1 44278071 EC50 = 180 nM T72458 C9Y7KM 44278193 EC50 = 13 nM T72458 CBWJ71 44278194 EC50 = 24 nM T72458 COS0B2 44278195 EC50 = 35 nM T72458 C8A1GE 44278223 EC50 = 130 nM T72458 CU0J1F 44279606 IC50 > 100000 nM T72458 CEG7U1 44279630 IC50 > 100000 nM T72458 CY9XO5 44279793 IC50 > 100000 nM T72458 CU8PH5 44293516 IC50 = 2.03 nM T72458 C7DZ1Q 44293599 EC50 = 3.38 nM T72458 C57HNX 44307979 IC50 > 10000 nM T72458 C8LZV7 44308004 IC50 > 10000 nM T72458 CFP7W8 44308044 IC50 > 10000 nM T72458 C79WRA 44308214 IC50 > 10000 nM T72458 CT76SR 44308215 IC50 > 10000 nM T72458 COY71H 44314826 EC50 = 0.17 nM T72458 CJAW38 44314951 IC50 > 10000 nM T72458 CA7B1G 44315095 IC50 = 9250 nM T72458 CPX2L1 44315335 IC50 > 10000 nM T72458 C3U0CW 44317053 EC50 = 1420 nM T72458 CKH3J2 44317070 EC50 = 3280 nM T72458 CAW8L7 44317241 EC50 = 20 nM T72458 CK7LG6 44317242 EC50 = 760 nM T72458 CZTI78 44317254 EC50 = 10 nM T72458 CVW5B7 44317276 EC50 = 70 nM T72458 C4ZST8 44317277 EC50 = 4800 nM T72458 C90PCI 44317278 EC50 = 1670 nM T72458 CLO83G 44317279 EC50 = 2500 nM T72458 CQ59BO 44320339 Ki = 1995.26 nM T72458 C6UML0 44322786 EC50 = 21.5 nM T72458 C3CL8S 44322787 EC50 = 6.3 nM T72458 C5SZ6K 44322788 EC50 = 38.5 nM T72458 C27QTD 44322795 EC50 = 1.6 nM T72458 C9HQ8Z 44322812 EC50 = 20.5 nM T72458 C3XED9 44322868 Ki = 220 nM T72458 C8P1HE 44322869 EC50 = 50 nM T72458 CJD5K7 44322895 EC50 = 11.5 nM T72458 CSH73B 44322896 EC50 = 4.6 nM T72458 C3V7PO 44322923 EC50 = 18 nM T72458 CA9F8I 44322924 EC50 = 53 nM T72458 C32ADM 44322957 EC50 = 22.5 nM T72458 CU1R6F 44322958 EC50 = 14.5 nM T72458 CPG80V 44322959 EC50 = 26.5 nM T72458 CJ73UR 44322977 EC50 = 16.5 nM T72458 CW5T8L 44322986 EC50 = 24 nM T72458 CN12SY 44322987 EC50 = 38.5 nM T72458 C8W2GN 44322994 EC50 = 42.5 nM T72458 CEV0F8 44323015 EC50 = 41 nM T72458 CSL38N 44323016 EC50 = 11 nM T72458 CEDS20 44323020 Ki = 57 nM T72458 CI70FV 44323029 Ki = 5 nM T72458 CNB32J 44323031 EC50 = 20 nM T72458 CP9FE1 44323032 EC50 = 13 nM T72458 CCX5N0 44323033 EC50 = 28 nM T72458 C7RT2W 44323034 EC50 = 21.3 nM T72458 CC9E1M 44323212 EC50 = 22 nM T72458 CX7H2C 44323233 Ki = 58 nM T72458 CW49BO 44323234 Ki = 87 nM T72458 C8BID0 44325926 IC50 = 38.7 nM T72458 C9MA4R 44343337 EC50 = 0.019 nM T72458 CD9ER8 44343341 IC50 = 1.8 nM T72458 C46OFK 44343362 EC50 = 0.573 nM T72458 CL8Y3V 44343363 EC50 = 0.018 nM T72458 CCLF38 44347081 Ki = 1300 nM T72458 CT5V4X 44347082 Ki = 3800 nM T72458 C0QW9K 44347105 Ki = 110 nM T72458 CWK01G 44347106 Ki = 58 nM T72458 C4Y2SW 44347107 Ki = 0.28 nM T72458 C60PGA 44347110 Ki = 960 nM T72458 CUEZ31 44347119 Ki = 0.37 nM T72458 CT03JB 44347219 Ki = 0.5 nM T72458 COD7W0 44347220 Ki = 0.26 nM T72458 CNP94O 44347221 Ki = 0.88 nM T72458 CBE37A 44347277 Ki = 4 nM T72458 CIZ30K 44347294 Ki = 4.3 nM T72458 C2YQM4 44347330 Ki = 3700 nM T72458 CX0Z1Y 44347331 Ki = 0.58 nM T72458 CAKI17 44347344 Ki = 0.06 nM T72458 CEIM86 44347370 Ki = 0.57 nM T72458 CS5ID0 44347378 Ki = 420 nM T72458 CDN35X 44347379 Ki = 600 nM T72458 CENG52 44347433 Ki = 1.6 nM T72458 CW1JY7 44347434 Ki = 0.096 nM T72458 C24GLU 44347435 Ki = 0.85 nM T72458 CSD69H 44347750 Ki = 1300 nM T72458 C1A6SC 44347765 Ki = 140 nM T72458 CY2K3L 44347766 Ki = 2000 nM T72458 C7U2KM 44347838 IC50 = 750 nM T72458 CK6FH3 44347927 IC50 = 3300 nM T72458 C2G4RI 44347976 Ki = 300 nM T72458 C9EA0M 44347977 Ki = 310 nM T72458 CN04GT 44347980 Ki = 180 nM T72458 CBW50H 44347987 Ki = 1500 nM T72458 CK93QZ 44347990 Ki = 670 nM T72458 C5BX1H 44348033 Ki = 2500 nM T72458 C27BLZ 44348035 Ki = 1600 nM T72458 CZ6R1G 44348039 Ki = 690 nM T72458 C4OS9M 44348046 Ki = 9300 nM T72458 C9JP8O 44348069 Ki = 270 nM T72458 CCI04W 44348070 Ki = 320 nM T72458 C58SIF 44348144 IC50 = 40000 nM T72458 CA4NE7 44348151 Ki = 620 nM T72458 CY96AB 44348152 Ki = 320 nM T72458 C0F1EA 44348183 EC50 > 10000 nM T72458 CC41MG 44348199 EC50 > 10000 nM T72458 CRSW34 44348200 EC50 = 6.3 nM T72458 CUM7X1 44348844 EC50 = 1000 nM T72458 C9I7PM 44348845 EC50 = 520 nM T72458 C3UWB5 44349006 EC50 = 1100 nM T72458 CT6G1M 44349008 EC50 = 2100 nM T72458 C6E7SA 44349019 EC50 = 24 nM T72458 CH4RT3 44349026 EC50 < 0.1 nM T72458 C6B2XF 44349055 EC50 = 110 nM T72458 CK7V8I 44349056 EC50 = 680 nM T72458 CDI5G1 44349057 EC50 = 470 nM T72458 CEB7L6 44349093 EC50 = 170 nM T72458 C17TCL 44349094 EC50 = 600 nM T72458 CZW0E4 44349105 EC50 = 4400 nM T72458 CC92YX 44349106 EC50 = 440 nM T72458 C84PZR 44349107 EC50 = 690 nM T72458 C8AT4B 44349110 EC50 = 1900 nM T72458 C2ZVP9 44349111 EC50 = 2400 nM T72458 C52OGQ 44349133 EC50 = 380 nM T72458 CZ36XH 44349134 EC50 = 2200 nM T72458 CY21EM 44349151 EC50 = 1600 nM T72458 CHP4U8 44349170 EC50 = 1000 nM T72458 C39SAR 44349173 EC50 = 5.2 nM T72458 C7RSC0 44349183 EC50 = 650 nM T72458 CWT14Q 44349221 IC50 = 3 nM T72458 CZ4M3J 44349222 IC50 = 3.3 nM T72458 CW9A4F 44349223 IC50 = 1.4 nM T72458 C7RMI0 44349224 IC50 = 11 nM T72458 CDW65K 44349226 IC50 = 220 nM T72458 CYHZ68 44349227 IC50 = 9.5 nM T72458 C3K9VR 44349228 IC50 = 19 nM T72458 C7OW3R 44349246 IC50 = 8.9 nM T72458 CBIV27 44349247 IC50 = 4.8 nM T72458 C8AU9D 44349461 EC50 = 530 nM T72458 C26WVI 44349469 IC50 = 13 nM T72458 CNYT90 44349470 IC50 = 32 nM T72458 C2XSM4 44349471 Ki = 2 nM T72458 CU9IJ2 44349593 EC50 = 83 nM T72458 CNB8U7 44349594 IC50 < 0.1 nM T72458 C6XV5P 44357167 IC50 = 12 nM T72458 CWBV76 44357280 IC50 = 22 nM T72458 C39OBA 44357294 IC50 = 18 nM T72458 CRP7I9 44357348 IC50 = 25 nM T72458 CG6HS3 44357406 IC50 = 21 nM T72458 C3TCL0 44357527 IC50 = 14 nM T72458 C3CX9P 44357528 IC50 = 110 nM T72458 CI3TO0 44357547 IC50 = 180 nM T72458 C2MFK4 44357575 IC50 = 90 nM T72458 C4QA0D 44357595 IC50 = 9 nM T72458 CH0XI2 44357626 IC50 = 22 nM T72458 CVZ1T6 44357786 IC50 = 10 nM T72458 C2MG1B 44358565 EC50 = 2.1 nM T72458 C8GKE0 44358566 EC50 = 820 nM T72458 C37KYE 44358608 IC50 = 2755 nM T72458 C7QTS9 44358609 EC50 = 500 nM T72458 CUH68B 44358622 IC50 = 9020 nM T72458 C6E9LI 44358625 IC50 = 5.598 nM T72458 C0WTS6 44358630 IC50 = 98 nM T72458 CN3EM4 44358633 IC50 = 3930 nM T72458 C8XY0P 44358639 IC50 = 2.27 nM T72458 C3TJC8 44358660 IC50 = 130 nM T72458 CM06ZW 44358669 IC50 = 2170 nM T72458 C2S6HF 44358693 IC50 = 2055 nM T72458 CQA6O7 44358695 EC50 > 5000 nM T72458 C81PLU 44358697 EC50 = 4050 nM T72458 CW8E5G 44358698 EC50 = 3060 nM T72458 CU89HD 44358705 EC50 = 260 nM T72458 C2VBG9 44358848 EC50 = 5800 nM T72458 C6RC5L 44358915 IC50 = 1197 nM T72458 CS0C2O 44358917 IC50 = 2990 nM T72458 C9ACB0 44360829 EC50 = 500 nM T72458 CX0ZW3 44361027 IC50 = 108 nM T72458 C2QW1I 44364160 IC50 = 45 nM T72458 CLMA12 44366081 IC50 = 0.23 nM T72458 C2DHN5 44366155 IC50 = 0.51 nM T72458 CYD6R3 44366171 IC50 = 0.5 nM T72458 CO7U1L 44366182 IC50 = 0.48 nM T72458 CL4CY1 44366187 IC50 = 270 nM T72458 C9JN3L 44366213 IC50 = 1.3 nM T72458 C36FMV 44366215 IC50 = 0.087 nM T72458 CS27ZR 44366381 IC50 = 0.16 nM T72458 C61CYL 44372908 EC50 = 77 nM T72458 CWT5B7 44372933 EC50 = 20 nM T72458 C8D1MC 44372942 EC50 = 1150 nM T72458 CEW35X 44372964 EC50 = 45 nM T72458 C2UCY5 44373177 EC50 = 20 nM T72458 CZ42QB 44373197 EC50 = 60 nM T72458 CCB05K 44373198 EC50 = 13 nM T72458 CX92FV 44373317 EC50 = 100 nM T72458 CR40BF 44383343 IC50 = 100 nM T72458 CQCP89 44387680 EC50 = 100 nM T72458 C7F3DV 44390411 EC50 = 4 nM T72458 CN3IE7 44390421 EC50 = 18 nM T72458 C5Y6HU 44390422 EC50 = 63 nM T72458 CR92QC 44390423 EC50 = 60 nM T72458 CEF15X 44390424 EC50 = 27 nM T72458 CP40IU 44391262 Ki = 110 nM T72458 CWO97F 44391271 Ki = 120 nM T72458 C58VDM 44391272 Ki = 160 nM T72458 CZMI04 44391285 Ki = 370 nM T72458 CGL71H 44391286 Ki = 270 nM T72458 C65PWK 44391288 Ki = 36 nM T72458 C9ZV5O 44391289 Ki = 110 nM T72458 CKT64C 44391303 Ki = 140 nM T72458 C1A6TX 44391304 Ki = 22 nM T72458 C07TBF 44391315 Ki = 41 nM T72458 CCV1R7 44391316 Ki = 87 nM T72458 C09FSO 44391379 Ki = 47 nM T72458 C0XPV5 44391380 Ki = 24 nM T72458 CVIE64 44391381 Ki = 120 nM T72458 CQU0T8 44391382 Ki = 10 nM T72458 CK7D6C 44391386 Ki = 52 nM T72458 C2B1EF 44391391 Ki = 56 nM T72458 C36DSN 44391402 Ki = 49 nM T72458 C0WT5A 44391403 Ki = 34 nM T72458 C39BFV 44391404 Ki = 33 nM T72458 CY8DP4 44391405 Ki = 30 nM T72458 CD8HL0 44392514 Ki = 860 nM T72458 CE21OM 44392535 Ki = 1500 nM T72458 C3IHV4 44393417 Ki = 390 nM T72458 C2J1ML 44393418 Ki = 1000 nM T72458 CQ3L0D 44393421 Ki = 1400 nM T72458 C9C7SD 44393430 Ki = 57000 nM T72458 C47HVD 44393441 Ki = 30000 nM T72458 C1OG5U 44393450 Ki = 169000 nM T72458 CX5F8Z 44393808 EC50 = 91 nM T72458 C3P9OV 44393809 EC50 = 36 nM T72458 CQ7ZW3 44393820 Ki = 84 nM T72458 CM1U6O 44393821 Ki = 35 nM T72458 CEX5T7 44393822 Ki = 24 nM T72458 C8NUV7 44393823 Ki = 145 nM T72458 CAT7F3 44393824 EC50 = 2.9 nM T72458 C6V0HU 44393850 EC50 = 40 nM T72458 CH60CQ 44393851 Ki = 49 nM T72458 CFJ6C3 44393862 Ki = 24 nM T72458 CZ2QV6 44393863 Ki = 25 nM T72458 CTM7X6 44393864 Ki = 13 nM T72458 CI8NO6 44393876 EC50 = 90 nM T72458 CI46JK 44393877 Ki = 102 nM T72458 CCV60F 44393885 EC50 = 18 nM T72458 CK2VD1 44393886 Ki = 23 nM T72458 C2IO4E 44393887 Ki = 11 nM T72458 CP8EQ1 44393888 Ki = 12 nM T72458 CR5BI0 44393889 Ki = 33 nM T72458 CN7YD9 44394009 Ki = 90 nM T72458 CS1YM0 44394010 Ki = 66 nM T72458 CKWJ51 44394078 Ki = 53 nM T72458 CK5D8I 44394079 Ki = 27 nM T72458 CT5C0V 44394080 Ki = 14 nM T72458 CM69EP 44394081 Ki = 81 nM T72458 C25TVF 44394093 EC50 = 168 nM T72458 C5K7CG 44394580 EC50 = 123 nM T72458 C08QML 44394581 EC50 = 38.5 nM T72458 C0OMU3 44394582 EC50 = 155 nM T72458 CL3P2Q 44394583 EC50 = 23.7 nM T72458 C5SGR6 44394584 EC50 = 150 nM T72458 CLXA10 44394585 EC50 = 13.7 nM T72458 C48NFW 44394586 EC50 = 68.7 nM T72458 C8GUD1 44394622 EC50 = 59.5 nM T72458 C9O4GM 44394623 EC50 = 4.6 nM T72458 C29ELZ 44394624 EC50 = 5 nM T72458 CP4A0B 44394625 EC50 = 88.5 nM T72458 C94PGA 44394626 EC50 = 159 nM T72458 CF4O9U 44394627 EC50 = 106 nM T72458 CZ37TO 44394654 EC50 = 39.3 nM T72458 CPE65R 44394655 EC50 = 35 nM T72458 C9LKB5 44394656 EC50 = 131 nM T72458 CG1Q8L 44394657 EC50 = 114 nM T72458 CHG12Y 44394658 EC50 = 31.3 nM T72458 C9OTX4 44394659 EC50 = 10.5 nM T72458 CNHD57 44394660 EC50 = 14.5 nM T72458 CHTM92 44394689 EC50 = 29.7 nM T72458 C04RCL 44394690 EC50 = 31.3 nM T72458 CT9D5Y 44394691 EC50 = 21 nM T72458 CHDB95 44394692 EC50 = 30 nM T72458 CHZF38 44394693 EC50 = 20 nM T72458 C9Y6ZI 44394694 EC50 = 121 nM T72458 C06PXF 44394695 EC50 = 82 nM T72458 CJ97VD 44394730 EC50 = 14.1 nM T72458 C1IE7P 44394731 EC50 = 8.5 nM T72458 CLF0X5 44394732 EC50 = 42 nM T72458 C9QR1L 44394733 EC50 = 12 nM T72458 CP1IR5 44394734 EC50 = 135 nM T72458 C2UY8G 44394735 EC50 = 18.7 nM T72458 CTY36S 44394736 EC50 = 27 nM T72458 CR5B6L 44394748 EC50 = 4527 nM T72458 CW13LR 44394749 EC50 = 137 nM T72458 CL3A0O 44394750 EC50 = 446 nM T72458 CIGZ40 44394783 EC50 = 45 nM T72458 C62FUR 44394784 EC50 = 58 nM T72458 CCZ37I 44394785 EC50 = 50 nM T72458 C8RHG3 44394786 EC50 = 96 nM T72458 CQD01R 44394787 EC50 = 185 nM T72458 CO43JY 44394788 EC50 = 146 nM T72458 CCE30Z 44394789 EC50 = 419 nM T72458 C8C6GY 44395416 Ki = 3900 nM T72458 CF3WX5 44395436 Ki = 600 nM T72458 C6ACZ4 44395464 Ki = 1000 nM T72458 CD6BN5 44395465 Ki = 3800 nM T72458 CS5O1J 44395466 Ki = 46 nM T72458 CC3Y5Q 44395503 Ki = 6400 nM T72458 CSAR32 44395513 Ki = 290 nM T72458 CAO42X 44395534 Ki = 5400 nM T72458 C8UY4T 44395535 Ki = 410 nM T72458 CQ7S4C 44395572 Ki = 1000 nM T72458 CSF9I6 44395614 Ki > 10000 nM T72458 C0S9PU 44395615 Ki = 30 nM T72458 C3T1KX 44395646 Ki = 1800 nM T72458 CA8M9V 44395647 Ki = 66 nM T72458 CP1K3Q 44395654 Ki = 38 nM T72458 CG1AR2 44395666 Ki > 10000 nM T72458 C9S6VA 44395667 Ki = 40 nM T72458 CVUQ61 44395681 Ki = 14 nM T72458 C6X2TM 44395869 Ki = 50 nM T72458 C1AN6P 44395899 Ki = 48 nM T72458 CAJM38 44395920 Ki = 140 nM T72458 C5VLQ9 44395948 Ki = 220 nM T72458 C35KSH 44395950 Ki = 26 nM T72458 CLT7X4 44396002 Ki = 41 nM T72458 CCZP29 44396036 Ki = 75 nM T72458 C0IF3K 44396067 Ki = 470 nM T72458 CR8UG7 44396068 Ki = 290 nM T72458 C6QME3 44396069 Ki = 430 nM T72458 C7QF9Y 44396079 Ki = 120 nM T72458 CJ39OH 44396102 Ki = 140 nM T72458 CYS89B 44396114 Ki = 110 nM T72458 C9TU4E 44396120 Ki = 86 nM T72458 C4NZF5 44396125 IC50 = 160 nM T72458 CLG84D 44396126 IC50 = 180 nM T72458 C63TUF 44396140 IC50 = 57.3 nM T72458 CPA70N 44396141 Ki = 210 nM T72458 CC15YA 44396158 Ki = 150 nM T72458 CQR2H1 44396953 Ki = 120 nM T72458 CN1SJ0 44396954 Ki = 270 nM T72458 C87ZDT 44396955 Ki = 340 nM T72458 CTNE47 44396956 Ki = 520 nM T72458 CZ59JV 44396957 Ki = 260 nM T72458 C8D2RU 44396986 EC50 = 238 nM T72458 C6Z9BD 44396987 IC50 = 14 nM T72458 C5OI8Q 44397027 Ki = 23 nM T72458 CZ2C9L 44397028 Ki = 7.6 nM T72458 C98DZS 44397029 Ki = 18 nM T72458 CDZ3O4 44397030 Ki = 8.4 nM T72458 CAZ6R7 44397053 Ki = 260 nM T72458 C34UVG 44397054 Ki = 490 nM T72458 CTF68U 44397079 Ki = 180 nM T72458 CZ7YU4 44397080 Ki = 340 nM T72458 CI8UE5 44397121 Ki = 61 nM T72458 CF6Z4Y 44397122 Ki = 92 nM T72458 CDS5M7 44397123 Ki = 110 nM T72458 CN83XR 44397124 Ki = 45 nM T72458 CI8H6N 44397125 Ki = 22 nM T72458 C6FXK8 44397129 Ki = 210 nM T72458 C4UNI8 44397130 Ki = 240 nM T72458 CK47TL 44397131 Ki = 250 nM T72458 CP9H1C 44397132 Ki = 350 nM T72458 CE1Y6G 44397133 Ki = 400 nM T72458 C7FG4M 44397195 Ki = 230 nM T72458 C9V2RU 44397198 Ki = 6.4 nM T72458 CSV12E 44397199 Ki = 21 nM T72458 CG0FU9 44397216 Ki = 290 nM T72458 C9CF7N 44397220 IC50 = 6 nM T72458 CPI0R3 44397222 Ki = 210 nM T72458 CIS6C5 44397223 Ki = 420 nM T72458 C25TBE 44397224 Ki = 36 nM T72458 C0BUD1 44397225 Ki = 62 nM T72458 CY4G9J 44397226 Ki = 540 nM T72458 CZV64D 44397279 Ki = 220 nM T72458 CU7E3B 44397280 Ki = 60 nM T72458 CXQ0M6 44397281 Ki = 11 nM T72458 CX2OM4 44397282 Ki = 18 nM T72458 CPM68W 44397283 Ki = 12 nM T72458 CX07ID 44397304 Ki = 12 nM T72458 C4ZE3U 44397307 Ki = 220 nM T72458 CV07QL 44397308 Ki = 190 nM T72458 CD81IL 44397337 IC50 = 1000 nM T72458 C32RCI 44397338 EC50 = 470 nM T72458 C5X6SW 44397339 IC50 = 290 nM T72458 C85BWQ 44397355 EC50 = 410 nM T72458 CYUE71 44397356 IC50 = 4.7 nM T72458 C7Z8GI 44397409 IC50 = 3.2 nM T72458 C7TNB6 44397410 EC50 = 61 nM T72458 CK6S9U 44397411 IC50 = 490 nM T72458 C3ODR7 44397412 EC50 = 550 nM T72458 C6XL4E 44397444 IC50 = 3.8 nM T72458 C40IAW 44397445 IC50 = 100 nM T72458 C6F0QR 44397455 IC50 = 0.56 nM T72458 CYF0K3 44397458 IC50 = 750 nM T72458 C8ZIU6 44397459 IC50 = 390 nM T72458 C30ZFY 44397460 IC50 = 160 nM T72458 C49FRZ 44397461 EC50 = 110 nM T72458 CFIQ85 44397534 EC50 = 1100 nM T72458 C4BWN8 44397535 IC50 = 1100 nM T72458 C2O0YK 44397569 EC50 = 210 nM T72458 C21NUS 44397570 EC50 = 680 nM T72458 CSI0J5 44397633 IC50 = 58 nM T72458 CD2ES6 44397651 IC50 = 36 nM T72458 CL6KA2 44397652 EC50 = 110 nM T72458 C78YOV 44397653 EC50 = 550 nM T72458 C3GM2K 44397654 EC50 = 710 nM T72458 C4OUF0 44397655 EC50 = 120 nM T72458 C3J8LY 44397657 EC50 = 200 nM T72458 C8H6EI 44397658 IC50 = 45 nM T72458 CQ6OU7 44397659 EC50 = 750 nM T72458 CIH93R 44397660 EC50 = 430 nM T72458 CKT12I 44397661 IC50 = 950 nM T72458 C1C8WZ 44397698 EC50 = 1100 nM T72458 CSYW04 44397700 IC50 = 17 nM T72458 CZJ60B 44397701 IC50 = 89 nM T72458 CRL32F 44397702 EC50 = 490 nM T72458 CNZ32D 44398259 EC50 = 19.95 nM T72458 C2YWK3 44398340 EC50 = 0.5012 nM T72458 CU7NG4 44400612 Ki = 23 nM T72458 CHGN15 44400658 Ki = 18 nM T72458 CJ36UT 44400660 Ki = 2.4 nM T72458 COM2E6 44400661 Ki = 3.1 nM T72458 C56OUG 44400662 Ki = 2 nM T72458 CTM72F 44400707 Ki = 18 nM T72458 C56BLV 44400708 Ki = 16 nM T72458 CL4A0W 44400709 Ki = 31 nM T72458 CQ8GK5 44400711 Ki = 14 nM T72458 COV9C6 44400768 Ki = 23 nM T72458 CJ4M7S 44400769 Ki = 420 nM T72458 CD4TC0 44400770 Ki = 5700 nM T72458 CO7NM3 44400777 Ki = 2.8 nM T72458 C0E3XG 44400778 Ki = 5 nM T72458 C0OC7A 44400809 Ki = 2.1 nM T72458 COJM70 44400810 Ki = 1.4 nM T72458 CFT4O6 44400811 Ki = 2.4 nM T72458 C5NJQ2 44400812 Ki = 5 nM T72458 CC8SI2 44400813 Ki = 2.9 nM T72458 C3I0DM 44400814 Ki = 1.3 nM T72458 C9SA2Y 44400824 Ki = 2300 nM T72458 C95VUG 44400825 Ki = 1100 nM T72458 C51RXY 44400834 Ki = 94 nM T72458 CAR95M 44400863 Ki = 4.5 nM T72458 C2VI7C 44400864 Ki = 1.7 nM T72458 CQ01GT 44400902 Ki = 3600 nM T72458 CQ16YO 44400903 Ki > 10000 nM T72458 C2MEL4 44400932 Ki = 4.6 nM T72458 C61RQJ 44400934 Ki = 2 nM T72458 C2IJZ5 44400935 Ki = 1.5 nM T72458 CYF7N9 44401275 Ki = 649 nM T72458 CKH54Y 44401285 Ki = 255 nM T72458 C1QM4Y 44401310 IC50 = 6 nM T72458 C1JK9O 44401341 Ki = 2780 nM T72458 CTOS16 44401367 Ki = 109 nM T72458 C3S2XK 44401371 Ki = 376 nM T72458 CH1OX7 44401386 Ki = 1057 nM T72458 CR8GT9 44401392 Ki = 8017 nM T72458 CBQ7N3 44401418 Ki = 667 nM T72458 C1O0YW 44401421 Ki > 50000 nM T72458 CJNH94 44401440 Ki = 138 nM T72458 CGA3W5 44401462 Ki > 50000 nM T72458 CUZJ52 44401513 Ki = 333 nM T72458 CM9W3D 44401520 EC50 = 5 nM T72458 CIQH79 44401522 EC50 = 3 nM T72458 CDSM37 44401524 EC50 = 5 nM T72458 CVN78D 44401528 IC50 = 5 nM T72458 C4R9XD 44401530 EC50 = 7 nM T72458 C9Y0LO 44401553 Ki = 47 nM T72458 C7E3YU 44401573 Ki = 1845 nM T72458 C5LID4 44401581 Ki = 310 nM T72458 C5AQD6 44401585 EC50 = 330 nM T72458 CGNC86 44401587 Ki = 10788 nM T72458 C74QHS 44401592 Ki = 243 nM T72458 CX30HI 44401607 Ki = 226 nM T72458 C1U3NV 44404522 EC50 = 3 nM T72458 CY80DJ 44404523 EC50 = 4 nM T72458 C5DB0V 44404524 EC50 = 6 nM T72458 C1CY7E 44404525 EC50 = 5 nM T72458 CUZ2B7 44404526 EC50 = 2 nM T72458 CNH3C0 44404528 EC50 = 130 nM T72458 C8RKY9 44404529 EC50 = 550 nM T72458 CNZL81 44404538 Ki = 472 nM T72458 CQC38R 44404540 Ki = 467 nM T72458 CKW61M 44404542 Ki = 261 nM T72458 CGT1S0 44404543 Ki = 157 nM T72458 C3LKV0 44404544 Ki = 106 nM T72458 CM2ER9 44404545 Ki = 125 nM T72458 C4MAJ1 44404546 Ki = 190 nM T72458 CVE9L3 44404547 Ki = 50 nM T72458 C72ONL 44404549 Ki = 14 nM T72458 C3F6JI 44404550 Ki = 111 nM T72458 CCF97M 44404560 Ki = 90 nM T72458 CW6UD5 44404561 Ki = 40 nM T72458 CUBW74 44404562 Ki = 130 nM T72458 CP7D1W 44404563 Ki = 110 nM T72458 CU92ZV 44404564 Ki = 40 nM T72458 C6QC2S 44404566 Ki = 150 nM T72458 C35QSF 44404567 Ki = 200 nM T72458 CPF03E 44404568 Ki = 70 nM T72458 CR93UF 44404570 Ki = 70 nM T72458 CKC91E 44404571 Ki = 20 nM T72458 CKY6G8 44404572 Ki = 190 nM T72458 C1TXF6 44404575 Ki = 150 nM T72458 C4IFA0 44404576 Ki = 100 nM T72458 C0FB6W 44404577 Ki = 483 nM T72458 C5EX1D 44404822 Ki = 900 nM T72458 CL8U6X 44404823 Ki = 900 nM T72458 CQMR23 44405360 Ki = 11 nM T72458 CGV7U9 44405361 Ki = 79 nM T72458 C3BP8S 44405362 Ki = 99 nM T72458 CN9FE0 44405364 Ki = 100 nM T72458 CJ95PM 44405365 Ki = 210 nM T72458 CX9E1R 44405366 Ki = 42 nM T72458 C4K9OG 44405368 Ki = 130 nM T72458 CA2D8P 44405374 Ki = 180 nM T72458 CD1U0B 44405375 Ki = 260 nM T72458 CK6S4G 44405376 Ki = 80 nM T72458 CMOH97 44405377 Ki = 120 nM T72458 CK36RZ 44405378 Ki = 140 nM T72458 CFW20E 44405382 Ki = 61 nM T72458 C8GE4Y 44405392 Ki = 280 nM T72458 CVF02W 44405395 Ki = 60 nM T72458 C8A0QP 44405402 Ki = 84 nM T72458 C75WLG 44405403 Ki = 97 nM T72458 CQK5O8 44405425 Ki = 82 nM T72458 CEVF76 44405426 Ki = 16 nM T72458 CSV9Z7 44405443 Ki = 170 nM T72458 CX1RP9 44405450 Ki = 100 nM T72458 C47ZWV 44405526 EC50 = 570 nM T72458 C7VJ2H 44405549 Ki = 140 nM T72458 CA21ST 44405553 Ki = 160 nM T72458 C9JUS5 44405558 Ki = 150 nM T72458 CXYL12 44405561 Ki = 270 nM T72458 CC68NS 44405562 Ki = 230 nM T72458 CUVK05 44405563 Ki = 1000 nM T72458 CF1W2D 44405582 Ki = 130 nM T72458 CH5BW3 44405596 Ki = 210 nM T72458 CVXJ50 44405613 Ki = 110 nM T72458 CB46SC 44405620 Ki = 300 nM T72458 C3NL7Z 44405681 EC50 = 3 nM T72458 C6TE2H 44405769 EC50 = 72 nM T72458 C5W2NU 44405770 EC50 = 5 nM T72458 CU3MJ7 44405773 EC50 = 2 nM T72458 CGMF87 44405785 EC50 = 50 nM T72458 CEH5M3 44405791 EC50 = 90 nM T72458 CRG17F 44405792 EC50 = 2 nM T72458 CA5N2U 44405793 EC50 = 2 nM T72458 CR9GY2 44405794 EC50 = 15 nM T72458 CYW82T 44405802 EC50 = 110 nM T72458 C2B0HL 44405812 EC50 = 5 nM T72458 C6YNC5 44405823 EC50 = 39 nM T72458 CKY6L1 44405825 EC50 = 85 nM T72458 CIY3N6 44405826 EC50 = 3 nM T72458 CH5E4L 44405832 EC50 = 200 nM T72458 CY63HS 44405833 EC50 = 2 nM T72458 CVHQ82 44405835 EC50 = 2 nM T72458 CT9WH8 44405836 EC50 = 2 nM T72458 C7FCD0 44405857 EC50 = 3 nM T72458 CMY9H2 44405858 EC50 = 2 nM T72458 C8AL0J 44405860 EC50 = 2 nM T72458 CL3T6Z 44405879 EC50 = 15 nM T72458 CDR54Z 44405910 EC50 = 2 nM T72458 C0H2SP 44405911 EC50 = 11 nM T72458 C4OM2E 44405913 EC50 = 220 nM T72458 CRMV98 44408154 EC50 = 5.8 nM T72458 CIWX60 44408155 IC50 = 2.1 nM T72458 COG72Y 44408173 EC50 = 5.3 nM T72458 C3CQ4J 44408189 IC50 = 4.3 nM T72458 CW08ZJ 44408190 IC50 = 4 nM T72458 CNWJ27 44408252 EC50 = 16 nM T72458 CH68SP 44408253 EC50 = 14 nM T72458 CCFV91 44408275 EC50 = 8.6 nM T72458 CZ3YG9 44408276 EC50 = 6.1 nM T72458 CAFP51 44408286 EC50 = 2.4 nM T72458 CR8HZ7 44408287 EC50 = 1.3 nM T72458 COC7D2 44408388 EC50 = 15 nM T72458 CJ4N3I 44409103 EC50 = 8 nM T72458 C2NJ0V 44409104 Ki = 13 nM T72458 CKF52N 44409140 EC50 = 160 nM T72458 C5XEI8 44409206 Ki = 76 nM T72458 C9EXZ2 44409337 EC50 = 38 nM T72458 CFT41O 44409338 Ki = 5 nM T72458 CUB1Q2 44409339 EC50 = 20 nM T72458 CK5GO1 44409379 EC50 = 193 nM T72458 CUD19G 44410040 Ki = 0.58 nM T72458 CH1E8N 44410041 Ki = 21 nM T72458 C4Y8LV 44410046 Ki = 26 nM T72458 C61ZVJ 44410175 Ki = 13 nM T72458 C06FAT 44410176 Ki = 2.8 nM T72458 COFW07 44410188 Ki = 5.1 nM T72458 C5QG1S 44410207 Ki = 700 nM T72458 C8F2TJ 44410349 Ki = 26000 nM T72458 CKRP65 44410378 Ki = 110 nM T72458 C6IB1X 44410379 Ki = 14 nM T72458 CL0H4T 44410385 Ki = 690 nM T72458 C48WZD 44410802 Ki = 17.3 nM T72458 C43IKV 44410803 Ki = 10.4 nM T72458 CC8DA0 44412509 Ki = 12 nM T72458 CX60PS 44412510 Ki = 10 nM T72458 C3KB7R 44412511 Ki = 148 nM T72458 C1EOW5 44412512 Ki = 26 nM T72458 CT2N0X 44412513 Ki = 3 nM T72458 C20OFY 44412559 Ki = 3427 nM T72458 C20ZDH 44412560 Ki = 4 nM T72458 CPQJ43 44412561 Ki = 4 nM T72458 CF5G4W 44412572 Ki = 326 nM T72458 C56OPH 44412574 Ki = 3 nM T72458 C9T3YV 44412612 Ki = 2 nM T72458 CSO69M 44412613 Ki = 10 nM T72458 CG23BY 44412626 Ki = 14 nM T72458 CJYM45 44412640 Ki = 13 nM T72458 CEK59C 44412641 Ki = 13 nM T72458 CB6K4I 44412642 Ki = 5 nM T72458 CRD87I 44412646 Ki = 18 nM T72458 CAF4V8 44412647 Ki = 35 nM T72458 CC2QB0 44412665 Ki = 54 nM T72458 CS8EC2 44412676 Ki = 1800 nM T72458 C1QPI3 44412677 Ki = 1500 nM T72458 CXNI74 44412678 Ki = 450 nM T72458 C3UF8S 44412679 Ki = 360 nM T72458 C1VA2R 44412680 Ki = 1000 nM T72458 C3Y0LF 44412681 Ki = 550 nM T72458 CZ3E0A 44412684 Ki = 1800 nM T72458 C65XZU 44412685 Ki = 440 nM T72458 C3GEM5 44412687 Ki = 1100 nM T72458 C57SDW 44412688 Ki = 1300 nM T72458 CLT8W2 44412690 Ki = 1000 nM T72458 CB6H8W 44412691 Ki = 560 nM T72458 C9K3XB 44412711 Ki = 2200 nM T72458 C6GO1C 44412729 Ki = 2600 nM T72458 C0NAS2 44412740 Ki = 1800 nM T72458 CE4QZ5 44412758 Ki = 7 nM T72458 C1K8LS 44412770 Ki = 2800 nM T72458 CX8K7T 44412791 Ki = 1200 nM T72458 CCZP41 44412864 Ki = 1200 nM T72458 CPU13S 44412869 Ki = 21 nM T72458 C9GRF4 44412881 Ki = 1300 nM T72458 CC49LZ 44412884 Ki = 130 nM T72458 C3Q6RO 44412896 Ki = 87 nM T72458 CNP17D 44412897 Ki = 12 nM T72458 CXDA47 44412898 Ki = 8.8 nM T72458 CF73OD 44412909 Ki = 420 nM T72458 CS02LO 44412910 Ki = 480 nM T72458 C6D3MA 44412911 Ki = 15 nM T72458 C7Z8WB 44412912 Ki = 180 nM T72458 CW31RQ 44412930 Ki = 200 nM T72458 CM1J9Q 44412931 Ki = 1500 nM T72458 C4KWB3 44412933 Ki = 1.6 nM T72458 CA9YQ3 44412963 Ki = 710 nM T72458 C0E7QK 44412964 Ki = 520 nM T72458 C0OWN7 44412990 Ki = 750 nM T72458 CA8BU2 44413002 Ki = 310 nM T72458 CJM74H 44413005 Ki = 170 nM T72458 CZX75O 44413056 Ki = 710 nM T72458 CW6ZC0 44413576 EC50 = 10133.6 nM T72458 CG59EP 44413600 Ki = 214.6 nM T72458 CZY3R6 44413602 Ki = 69.6 nM T72458 CJ71PZ 44413604 Ki = 369.9 nM T72458 CPB02M 44413606 Ki = 41.8 nM T72458 CHT0V3 44413652 Ki = 43.9 nM T72458 C0AT2B 44413666 Ki = 68.4 nM T72458 CJY9Q1 44413668 Ki = 5 nM T72458 CN3WD2 44413684 Ki = 100.7 nM T72458 CJQ3N4 44413687 Ki = 46.9 nM T72458 C4T2ES 44413741 Ki = 37.5 nM T72458 C24AUD 44413828 EC50 = 36 nM T72458 C08PBM 44413829 EC50 = 54 nM T72458 CT4FW5 44413830 EC50 = 8 nM T72458 C8IDV1 44413831 EC50 = 457 nM T72458 CZ3Q4T 44413832 EC50 = 515 nM T72458 CV6Z8C 44413842 EC50 = 1617 nM T72458 C4P0LS 44413879 EC50 = 152 nM T72458 C84OJQ 44413880 EC50 = 249 nM T72458 CN7I2S 44413881 EC50 = 254 nM T72458 CF6O4K 44413913 EC50 = 184 nM T72458 CS42BM 44413914 EC50 = 3.7 nM T72458 CN18BL 44413930 EC50 = 14 nM T72458 C4BMF6 44413931 EC50 = 4.3 nM T72458 C9WNH8 44413932 EC50 = 17 nM T72458 CKZ86P 44413938 EC50 = 20 nM T72458 CL2RK9 44413968 EC50 = 1093 nM T72458 CM2J9Z 44413969 Ki = 1712 nM T72458 C34XGB 44413970 Ki = 6666 nM T72458 CA5K6H 44415336 Ki > 10000 nM T72458 CW4FC2 44415337 Ki = 2600 nM T72458 CEU1V2 44415346 Ki = 86 nM T72458 CJ81VG 44415347 Ki = 4000 nM T72458 CDJ81P 44415348 Ki > 10000 nM T72458 CJ3K6S 44415359 Ki = 57 nM T72458 CJ74MF 44415360 Ki = 2500 nM T72458 CS4D9A 44415361 Ki = 350 nM T72458 CW25PK 44415369 Ki = 2800 nM T72458 CIA0T1 44415370 Ki = 1700 nM T72458 C2YMO0 44415377 Ki = 300 nM T72458 CEW9H0 44415384 Ki = 3300 nM T72458 CA8P2G 44415388 Ki = 400 nM T72458 CHC07X 44415398 Ki = 210 nM T72458 CX2WN0 44415405 Ki = 75 nM T72458 CC29YV 44415406 Ki = 74 nM T72458 C7IYH9 44415417 Ki = 110 nM T72458 C0QMO7 44415418 Ki = 94 nM T72458 CV2UY4 44415429 Ki = 690 nM T72458 CY8F9L 44415430 Ki = 1000 nM T72458 CEG71C 44415433 Ki = 140 nM T72458 C01ZBF 44415434 Ki = 170 nM T72458 CHK45T 44415442 Ki = 620 nM T72458 C1B6CI 44415453 Ki = 160 nM T72458 CECU63 44415479 Ki = 25 nM T72458 C6YI9R 44415521 Ki = 490 nM T72458 CKX67G 44415522 Ki = 190 nM T72458 CZ48AF 44415537 Ki = 1400 nM T72458 C84OHY 44415545 Ki = 2100 nM T72458 C2NQ3C 44415546 Ki = 2200 nM T72458 C4ERO9 44415630 Ki = 56 nM T72458 C7Z3YB 44415631 Ki = 1800 nM T72458 C24YUZ 44415659 Ki = 89 nM T72458 C1C2GZ 44415660 Ki = 2400 nM T72458 CGR80P 44415674 Ki = 110 nM T72458 CV0TQ9 44415675 Ki = 360 nM T72458 C6YM0F 44415691 Ki = 2800 nM T72458 CAH6W2 44415692 Ki = 64 nM T72458 CKWO35 44415693 Ki = 18 nM T72458 CT0A3Y 44415706 Ki = 780 nM T72458 C1MG0H 44415707 Ki = 30 nM T72458 C07BZO 44415709 Ki = 1900 nM T72458 CYC49B 44415725 Ki = 4600 nM T72458 C10ZBJ 44415726 Ki = 2300 nM T72458 C5BIZ4 44415727 Ki = 5900 nM T72458 CZ63NT 44415746 Ki = 4900 nM T72458 CBYA87 44415747 Ki = 640 nM T72458 CTEW36 44415748 Ki = 3000 nM T72458 C3F2MN 44415764 Ki = 2600 nM T72458 CQ4C0E 44415765 Ki = 1500 nM T72458 CNR4B5 44415766 Ki = 1600 nM T72458 C9L1FV 44415767 Ki = 92 nM T72458 CM0UP6 44415790 Ki = 4300 nM T72458 CKB35A 44415791 Ki = 2500 nM T72458 CWK5C9 44415809 Ki = 6100 nM T72458 C8Y2QU 44415902 Ki = 820 nM T72458 C3KQ8H 44415912 EC50 = 1.6 nM T72458 CDN97X 44415913 EC50 = 0.3 nM T72458 CAL83K 44415914 EC50 = 0.2 nM T72458 C5CF0M 44415918 EC50 = 2 nM T72458 CXI18W 44415919 Ki = 0.4 nM T72458 C6DH7I 44415920 Ki = 1.3 nM T72458 CIM96K 44415925 Ki = 1100 nM T72458 C1X0OG 44415926 Ki = 5700 nM T72458 C9GO0A 44415940 Ki = 4100 nM T72458 CL95SI 44415941 Ki = 4200 nM T72458 C06CYU 44415956 EC50 = 809 nM T72458 C76IXM 44415961 Ki > 10000 nM T72458 CE24IH 44415965 Ki = 47 nM T72458 C6KGF3 44415966 Ki = 31 nM T72458 CD2A9T 44415972 EC50 = 140 nM T72458 CP0GH2 44415984 Ki = 120 nM T72458 CA7YJ4 44415985 Ki = 920 nM T72458 CHT4E8 44415991 EC50 = 45 nM T72458 CHJ4T5 44416006 Ki = 3100 nM T72458 CV42LA 44416007 Ki = 2200 nM T72458 CPX62S 44416014 EC50 = 18 nM T72458 C6CHM0 44416020 Ki = 2800 nM T72458 CQ7P9R 44416023 Ki = 4500 nM T72458 C4HU5K 44416024 Ki = 4000 nM T72458 CB6Y3A 44416025 Ki = 1500 nM T72458 CITW80 44416043 Ki = 2500 nM T72458 CX12AI 44416044 Ki = 2500 nM T72458 CXNE97 44416045 Ki = 3600 nM T72458 C8A5KJ 44416046 Ki = 2100 nM T72458 C69CUX 44416057 EC50 = 0.34 nM T72458 C56DHI 44416060 EC50 = 1.6 nM T72458 C0LIB3 44416071 Ki = 2900 nM T72458 CZ78QT 44416072 Ki = 2600 nM T72458 C05WHL 44416073 Ki = 2000 nM T72458 C8PA7D 44416074 Ki = 4800 nM T72458 C14XFK 44416075 Ki > 10000 nM T72458 CJI3N4 44416092 Ki = 4400 nM T72458 CK35LI 44416093 Ki = 3800 nM T72458 CS0JZ7 44416094 Ki > 10000 nM T72458 CB2TU4 44416106 EC50 = 0.5 nM T72458 C6Y3SN 44416108 Ki = 4600 nM T72458 CY12SN 44416109 Ki = 3100 nM T72458 CP9T4B 44416122 EC50 = 12 nM T72458 C4FI3Y 44416126 Ki = 2600 nM T72458 C9KLB0 44416135 EC50 = 2.2 nM T72458 C37XPA 44416152 Ki = 5.3 nM T72458 CB3WH4 44416160 Ki = 60 nM T72458 CE32FW 44416161 Ki = 38 nM T72458 C8IFH0 44416162 Ki = 67 nM T72458 CT89FC 44416163 Ki = 160 nM T72458 CC93LB 44416182 Ki = 36 nM T72458 CWF02K 44416183 Ki = 8.8 nM T72458 CI4EV8 44416184 Ki = 80 nM T72458 CWE8T7 44416194 Ki = 71 nM T72458 CE1FA5 44416197 Ki = 6.5 nM T72458 C74NDV 44416200 Ki = 67 nM T72458 CRYG36 44416201 Ki = 16 nM T72458 C53WDB 44416208 Ki = 240 nM T72458 CSM1D2 44416209 Ki = 200 nM T72458 CZ7M5G 44416213 Ki = 12 nM T72458 C0YN8C 44416214 Ki = 1700 nM T72458 CN38JL 44416227 Ki = 230 nM T72458 CD4B9L 44416228 Ki = 120 nM T72458 C1NMV4 44416251 Ki = 92 nM T72458 CF4GR8 44416286 Ki = 5.9 nM T72458 CFKR01 44416298 Ki = 20 nM T72458 CTB6N2 44416299 Ki = 8.1 nM T72458 C9EVI6 44416327 Ki = 9.1 nM T72458 CTZ02S 44416338 Ki = 390 nM T72458 C9AUM3 44416349 Ki = 31 nM T72458 CI1A0C 44416361 Ki = 26 nM T72458 CU7C3F 44416375 Ki = 140 nM T72458 C7SC9P 44417549 IC50 = 1.8 nM T72458 CBCR82 44417551 IC50 = 4.1 nM T72458 CK0P4I 44417552 IC50 = 0.7 nM T72458 CT58RV 44417554 IC50 = 101 nM T72458 C32QEO 44418413 EC50 > 10000 nM T72458 C7FEU6 44418420 EC50 > 10000 nM T72458 CZW07E 44418421 EC50 > 10000 nM T72458 CLQG83 44418430 EC50 = 2.7 nM T72458 C8VG1S 44418431 IC50 = 1.2 nM T72458 C3HPI5 44418437 EC50 > 10000 nM T72458 CMD5N2 44418438 EC50 > 10000 nM T72458 CQE30X 44422937 IC50 = 1600 nM T72458 C6H0NU 44422958 IC50 > 10000 nM T72458 C7I0KW 44422959 IC50 > 10000 nM T72458 C46XOB 44422960 IC50 > 10000 nM T72458 CNM90E 44422961 IC50 > 10000 nM T72458 C2LQW9 44422997 IC50 = 4500 nM T72458 CJM09S 44422998 IC50 = 3600 nM T72458 CI9HF1 44422999 IC50 = 1200 nM T72458 CXH5F8 44423009 IC50 = 590 nM T72458 C3VOD0 44423010 IC50 = 4800 nM T72458 C7UI3W 44423011 IC50 > 5000 nM T72458 CI05BD 44423012 IC50 > 10000 nM T72458 C5EJ3P 44423013 IC50 > 10000 nM T72458 C2NR7G 44423014 IC50 > 10000 nM T72458 C3I2NF 44423359 IC50 = 333 nM T72458 CBDI21 44423373 IC50 = 52.7 nM T72458 CY73KM 44423376 IC50 = 52.2 nM T72458 CB3M0V 44423378 IC50 = 18.3 nM T72458 COZ8M7 44423380 IC50 = 98.6 nM T72458 C9OGJ7 44423382 IC50 = 23.4 nM T72458 C0U7DO 44423384 IC50 = 14.5 nM T72458 C8GO6W 44423420 IC50 = 594 nM T72458 CVSF54 44423421 IC50 = 567 nM T72458 CEH52R 44423422 IC50 = 208 nM T72458 C4MO9L 44423424 IC50 = 218 nM T72458 C02WHJ 44423425 IC50 = 341 nM T72458 CA01NG 44423426 IC50 = 1250 nM T72458 CXA18B 44423427 IC50 = 1870 nM T72458 C17DFM 44423428 IC50 = 1190 nM T72458 C7EM3T 44423429 IC50 = 336 nM T72458 CP8BY0 44423430 IC50 = 105 nM T72458 CB6JP2 44423431 IC50 = 177 nM T72458 CE8U4Y 44423432 IC50 = 147 nM T72458 CV53RU 44423433 IC50 = 241 nM T72458 C40UAO 44423434 IC50 > 10000 nM T72458 C6JZ4Q 44423435 IC50 = 745 nM T72458 C36BEG 44423436 IC50 = 653 nM T72458 C58ZAM 44423437 IC50 = 132 nM T72458 C3KQR1 44423438 IC50 = 2300 nM T72458 C0OA8S 44423439 IC50 = 565 nM T72458 CBI7U4 44423440 IC50 = 159 nM T72458 CMNR76 44423441 IC50 = 296 nM T72458 CF6SQ1 44423442 IC50 = 226 nM T72458 CB46XE 44423443 IC50 = 756 nM T72458 CC3VY2 44423444 IC50 = 36.8 nM T72458 C8RX6Y 44423445 IC50 = 228 nM T72458 CC9GO8 44423446 IC50 = 26 nM T72458 C3S7UM 44423447 IC50 = 82.8 nM T72458 CDP0C8 44423448 IC50 = 47.2 nM T72458 CQCX97 44423449 IC50 = 18 nM T72458 CQ4DG9 44423450 IC50 = 186 nM T72458 C1CZK0 44423451 IC50 = 65.1 nM T72458 C6S4WV 44423452 IC50 = 156 nM T72458 C3J0ZH 44423453 IC50 = 243 nM T72458 CK8TR1 44423454 IC50 = 23 nM T72458 CNB0L9 44423455 IC50 = 33 nM T72458 C8FBW9 44423456 IC50 = 27.1 nM T72458 CV54PE 44423457 IC50 = 11.7 nM T72458 CG45MD 44423458 IC50 = 27.1 nM T72458 CM0K5Y 44423459 IC50 = 24.3 nM T72458 CFLS73 44423460 IC50 = 15.2 nM T72458 CX2T9W 44423461 IC50 = 36.8 nM T72458 C6D1CU 44423462 IC50 = 23.6 nM T72458 CR3XM9 44423463 IC50 = 10.5 nM T72458 C93PXI 44423464 IC50 = 53.2 nM T72458 C1UI9Z 44423465 IC50 = 41.8 nM T72458 C1WX7C 44423466 IC50 = 42.6 nM T72458 C80QNR 44423467 IC50 = 100 nM T72458 CAU4H2 44423468 IC50 = 228 nM T72458 C3Y0VW 44423469 IC50 = 62.8 nM T72458 CW78PM 44423470 IC50 = 85.9 nM T72458 CN07QR 44423471 IC50 = 92.5 nM T72458 CNKS25 44426649 IC50 = 900 nM T72458 CN5RD6 44431510 EC50 > 10000 nM T72458 CF3H8A 44431511 EC50 > 10000 nM T72458 CVB07O 44431512 EC50 = 3200 nM T72458 CY80GN 44431513 IC50 = 1700 nM T72458 COCE51 44431515 EC50 = 2.87 nM T72458 CIM51K 44432885 Ki = 1000 nM T72458 CJN61T 44432891 Ki = 17000 nM T72458 C2W8XE 44432895 Ki = 11000 nM T72458 CI1Y8B 44432897 Ki = 630.96 nM T72458 CV03FK 44432898 Ki = 60 nM T72458 COW1J6 44432899 Ki = 218.78 nM T72458 CC0AJ8 44432900 Ki = 128.82 nM T72458 CLH19Y 44432902 Ki = 51 nM T72458 C4E2AY 44432903 Ki = 11.75 nM T72458 CZ3DA9 44432906 Ki = 7.9 nM T72458 C2C0YT 44432909 Ki = 4.898 nM T72458 CI61RS 44432913 Ki = 32.36 nM T72458 CPBJ64 44432916 Ki = 724.44 nM T72458 CC1FG7 44432917 Ki = 50 nM T72458 CABP12 44432918 Ki > 10000 nM T72458 CRHG83 44432920 Ki = 2290.87 nM T72458 CWF23Z 44432924 Ki = 4.467 nM T72458 CAK9Z8 44432927 Ki = 109.65 nM T72458 CWV84F 44432928 Ki = 7.244 nM T72458 CXPZ80 44432930 Ki = 5 nM T72458 CNM17K 44432931 Ki = 2.692 nM T72458 CV62SP 44432932 Ki = 3.3 nM T72458 CP1G3N 44432933 Ki = 6.457 nM T72458 CDHA64 44432939 Ki = 3.7 nM T72458 C7DZ3N 44432941 Ki = 0.8913 nM T72458 CPG0Z7 44432943 Ki = 2.138 nM T72458 CO7D3R 44432945 Ki = 8.3 nM T72458 CSM8T7 44432946 Ki = 8.71 nM T72458 CGNI61 44432947 Ki = 7.5 nM T72458 CD0ZV7 44432948 Ki = 5.2 nM T72458 C5P1UZ 44432949 Ki = 2.042 nM T72458 CVX47L 44432950 Ki = 1.7 nM T72458 CC06WF 44432951 Ki = 9.7 nM T72458 CHQO21 44432952 Ki = 4.169 nM T72458 CB62YF 44432953 Ki = 14 nM T72458 C2N0MD 44432954 Ki = 33 nM T72458 C0EY7P 44432955 Ki = 17.38 nM T72458 CX3NB9 44432956 Ki = 5.754 nM T72458 C3P5QE 44432957 Ki = 30.9 nM T72458 CXP4J8 44432958 Ki = 77.62 nM T72458 CKNT36 44432959 Ki = 19.95 nM T72458 C0V2US 44432960 Ki = 44.67 nM T72458 CN41MP 44432962 Ki = 3.2 nM T72458 CBRG36 44432963 Ki = 2.9 nM T72458 CL3ZR1 44432964 Ki = 3.89 nM T72458 CDNP90 44432965 Ki = 28 nM T72458 C0L4NV 44432966 Ki = 0.955 nM T72458 CW6V3C 44433158 Ki = 770 nM T72458 C3B7EG 44433262 Ki = 6.4 nM T72458 CPRL53 44433263 Ki = 26 nM T72458 CKX7P2 44433264 Ki = 4.5 nM T72458 CQ91YU 44433265 Ki = 6.2 nM T72458 CJZ3P7 44433266 Ki = 7.9 nM T72458 CRP35K 44433267 Ki = 6.4 nM T72458 CF3J7G 44433268 Ki = 8.7 nM T72458 C3ZIE0 44433269 Ki = 60 nM T72458 CN51TW 44433270 Ki = 1 nM T72458 CQ4X7E 44433271 Ki = 1.5 nM T72458 C4O5HS 44433272 Ki = 3.8 nM T72458 CEA96F 44433273 Ki = 49 nM T72458 CED62W 44433274 Ki = 120 nM T72458 CI29CM 44433275 Ki = 56 nM T72458 CEN1M3 44433276 Ki = 0.95 nM T72458 C9KT3N 44433277 Ki = 1.4 nM T72458 CS2YQ7 44433278 Ki = 140 nM T72458 C27GZL 44433279 Ki = 27 nM T72458 CB29IZ 44433282 Ki = 240 nM T72458 COX3A0 44433283 Ki = 40 nM T72458 CAE5J2 44433284 Ki = 3.8 nM T72458 C9U4FM 44433285 Ki = 2.4 nM T72458 CB6P5W 44433286 Ki = 6 nM T72458 C3R0EA 44433287 Ki = 1 nM T72458 CZN71T 44433288 Ki = 23 nM T72458 CR54CU 44433289 Ki = 7 nM T72458 C1M0JP 44433290 Ki = 0.71 nM T72458 C9ZT8U 44433291 Ki = 26 nM T72458 CI62TG 44433292 Ki = 57 nM T72458 CZ3I4N 44433293 Ki = 2 nM T72458 CZU4D1 44433294 Ki = 1.9 nM T72458 CS5TK4 44433295 Ki = 5 nM T72458 CYH7M2 44433296 Ki = 1.1 nM T72458 C7E4KR 44433297 Ki = 2.6 nM T72458 CPX57U 44433298 Ki = 1.4 nM T72458 CI2PC5 44433299 Ki = 1.5 nM T72458 C89WJP 44433300 Ki = 12 nM T72458 CEJ6Q8 44433378 Ki = 82 nM T72458 CYHD52 44433379 Ki = 390 nM T72458 C16UBL 44433380 Ki = 66 nM T72458 C1ABU5 44433381 Ki = 30 nM T72458 CUX68D 44433382 Ki = 96 nM T72458 CF3GN1 44433383 Ki = 95 nM T72458 C6Z9HA 44433384 Ki = 26 nM T72458 CG9N7V 44433385 Ki = 120 nM T72458 CVB59A 44433386 Ki = 180 nM T72458 CMH6O4 44433387 Ki = 260 nM T72458 C92BPS 44433388 Ki = 67 nM T72458 CC7VN4 44433389 Ki = 110 nM T72458 CTZI97 44433391 Ki = 59 nM T72458 CVX59F 44433392 Ki = 68 nM T72458 CHS4F5 44433406 Ki = 78 nM T72458 CNY6A2 44433407 Ki = 75 nM T72458 CLD9V1 44433409 Ki = 100 nM T72458 CW7SE3 44433411 Ki = 65 nM T72458 CJ20VN 44433413 Ki = 220 nM T72458 C39SZC 44433417 Ki = 31 nM T72458 CAZI23 44433418 Ki = 260 nM T72458 C6JPQ5 44433419 Ki = 250 nM T72458 CEGB56 44433420 Ki = 540 nM T72458 CFL4Z1 44433421 Ki = 350 nM T72458 CUM4N7 44433422 Ki = 160 nM T72458 C06KHC 44433423 Ki = 12 nM T72458 CG6O4A 44433424 Ki = 64 nM T72458 CKG92E 44433425 Ki = 200 nM T72458 CA6Z1R 44433426 Ki = 6.6 nM T72458 CTKI96 44433428 Ki = 12 nM T72458 CW8B6E 44433439 Ki = 8.6 nM T72458 C59IFV 44433441 Ki = 36 nM T72458 CI47FK 44433442 Ki = 15 nM T72458 CHG0X4 44433444 Ki = 18 nM T72458 CLJ9O6 44433445 Ki = 18 nM T72458 CZ7A5U 44433446 Ki = 5.4 nM T72458 C2T3MY 44433448 Ki = 21 nM T72458 C0OZ2S 44433450 Ki = 580 nM T72458 C7H8YL 44433455 Ki = 205 nM T72458 CO13HI 44433475 Ki = 43 nM T72458 C8NU0W 44433478 Ki = 81 nM T72458 CJ2D4S 44433479 Ki = 32 nM T72458 C5X8MW 44433480 Ki = 26 nM T72458 C9OZF5 44433481 Ki = 9.3 nM T72458 CAD9F7 44433482 Ki = 94 nM T72458 CH3KR5 44433483 Ki = 340 nM T72458 CQI17F 44433484 Ki = 98 nM T72458 C68VOP 44433561 Ki = 74 nM T72458 CYCP31 44433562 Ki = 26 nM T72458 CTF0P5 44433563 Ki = 4.5 nM T72458 CZQ3I4 44433564 Ki = 610 nM T72458 CLQI91 44434545 Ki = 39 nM T72458 C6DK3A 44434546 Ki = 1.8 nM T72458 C70WCO 44434547 Ki = 1.8 nM T72458 C2DH7G 44434548 Ki = 1 nM T72458 CHU9Q7 44434549 Ki = 10 nM T72458 C28NVB 44434550 Ki = 0.8 nM T72458 C4KQ0A 44434551 Ki = 26 nM T72458 C9M2BQ 44434552 Ki = 47 nM T72458 CVW3Q1 44434553 Ki = 3.3 nM T72458 CD5G6X 44434554 Ki = 49 nM T72458 CKN63U 44434555 Ki = 2.5 nM T72458 C52DTH 44434556 Ki = 29 nM T72458 C2WS3C 44434557 Ki = 7.5 nM T72458 CX6KL8 44434558 Ki = 6 nM T72458 CA39RJ 44434559 Ki = 3.3 nM T72458 C8HG1P 44434560 Ki = 7.1 nM T72458 C8Z1IM 44434561 Ki = 78000 nM T72458 C5C6IA 44434562 Ki = 0.8 nM T72458 CCP2N5 44434563 Ki = 2.3 nM T72458 C6KPV5 44434568 Ki = 4.5 nM T72458 C2K9TI 44434570 Ki = 106000 nM T72458 CKL0H4 44434572 Ki = 5800 nM T72458 CO0N2A 44434575 Ki = 8.8 nM T72458 CRJN03 44434579 Ki = 38 nM T72458 CKI3L6 44434580 Ki = 21000 nM T72458 CBC27H 44434581 Ki = 10000 nM T72458 C51NSB 44434584 Ki = 4900 nM T72458 CF2S6P 44434587 Ki = 2400 nM T72458 CQ81UI 44434592 Ki = 19000 nM T72458 CP2A4G 44434595 Ki = 9800 nM T72458 CT20IC 44434597 Ki = 164000 nM T72458 CC1H3U 44434598 Ki = 32000 nM T72458 CH17AO 44434599 Ki = 23000 nM T72458 CAID38 44434600 Ki = 81000 nM T72458 CGN1P8 44434601 Ki = 6400 nM T72458 CDV61Y 44434603 Ki = 7000 nM T72458 CZPC57 44434605 Ki = 14000 nM T72458 C5DT7Q 44434611 Ki = 11000 nM T72458 C3MS2D 44434613 Ki = 21000 nM T72458 C5A1GF 44434614 Ki = 16000 nM T72458 CN4D2E 44434616 Ki = 158000 nM T72458 C1B5RV 44434621 Ki = 10000 nM T72458 C5TMA6 44434625 Ki = 222000 nM T72458 C9XG2K 44434631 Ki = 165000 nM T72458 CY2C7G 44434632 Ki = 18000 nM T72458 CQ94YK 44434633 Ki = 5400 nM T72458 CM1NA8 44434634 Ki = 7100 nM T72458 C93NCL 44434635 Ki = 17000 nM T72458 CZ8TO1 44434636 Ki = 6200 nM T72458 CQ06DV 44434637 Ki = 77000 nM T72458 C0SM2J 44434647 Ki = 14000 nM T72458 C9GIF5 44434648 Ki = 9400 nM T72458 CTQ16K 44434649 Ki = 8400 nM T72458 C15MAF 44434650 Ki = 8100 nM T72458 CWD27I 44434651 Ki = 7100 nM T72458 C6X8WB 44434652 Ki = 16000 nM T72458 CWU74N 44434653 Ki = 2300 nM T72458 CXN0M3 44434654 Ki = 59000 nM T72458 CM0VZ8 44434655 Ki = 4700 nM T72458 CP0V1N 44434656 Ki = 99000 nM T72458 CV5Y3N 44434657 Ki = 13000 nM T72458 CVC93Q 44434658 Ki = 21000 nM T72458 CWE1V4 44434659 Ki = 96000 nM T72458 C5WR3A 44434661 Ki = 14000 nM T72458 CJ27QL 44434662 Ki = 6400 nM T72458 C6US7A 44434663 Ki = 5000 nM T72458 C4ZD1B 44434664 Ki = 87000 nM T72458 C03NKU 44434665 Ki = 44000 nM T72458 CJ2AT0 44434666 Ki = 5900 nM T72458 CF41SX 44434682 Ki = 3800 nM T72458 C9IWD4 44434683 Ki = 11000 nM T72458 CJ03PB 44434684 Ki = 3400 nM T72458 CIH0Z6 44434685 Ki = 3700 nM T72458 C4POB8 44434686 Ki = 9800 nM T72458 C1GFE6 44434687 Ki = 7400 nM T72458 C3J7WI 44434688 Ki = 3800 nM T72458 C9Y0BM 44434689 Ki = 17000 nM T72458 CH6LA5 44434690 Ki = 2000 nM T72458 CPRE40 44434691 Ki = 3700 nM T72458 C9O8LX 44434692 Ki = 2400 nM T72458 CE2Z3V 44434693 Ki = 2100 nM T72458 C31LUY 44434694 Ki = 2100 nM T72458 C9C4BN 44434695 Ki = 3700 nM T72458 CF3JX5 44434696 Ki = 1500 nM T72458 CM51SC 44434697 Ki = 2200 nM T72458 CA2FQ4 44434698 Ki = 2700 nM T72458 CTC18P 44434699 Ki = 4300 nM T72458 CQT85W 44434700 Ki = 4500 nM T72458 C8BQ7C 44434701 Ki = 3000 nM T72458 CV2QW3 44434702 Ki = 3400 nM T72458 C9IY3A 44434703 Ki = 2300 nM T72458 CF8J2P 44434704 Ki = 4100 nM T72458 CH7QD5 44434706 Ki = 2100 nM T72458 CT4FO2 44434707 Ki = 1900 nM T72458 C9E4PO 44434709 Ki = 4400 nM T72458 C7LUV2 44434713 Ki = 4100 nM T72458 CR70OD 44434714 Ki = 5600 nM T72458 CA1BF3 44434715 Ki = 4800 nM T72458 C0N4CY 44434753 Ki = 2500 nM T72458 CS1KG4 44434754 Ki = 6400 nM T72458 C2JHP0 44434757 Ki = 3200 nM T72458 CZ43DV 44434758 Ki = 1300 nM T72458 C50PIJ 44434759 Ki = 5600 nM T72458 CKAQ59 44434760 Ki = 2800 nM T72458 CALF38 44434761 Ki = 14000 nM T72458 C17HCY 44434762 Ki = 1500 nM T72458 CX75CS 44434763 Ki = 1900 nM T72458 CNB68V 44434764 Ki = 2300 nM T72458 CZ0R9M 44434765 Ki = 1900 nM T72458 CU9C0K 44434766 Ki = 1600 nM T72458 C8IHB1 44434767 Ki = 2400 nM T72458 C27KYV 44434768 Ki = 2600 nM T72458 CEM27N 44434769 Ki = 5300 nM T72458 CB7A2G 44434770 Ki = 3000 nM T72458 C0Y3IG 44434771 Ki = 3000 nM T72458 CNL2T3 44434772 Ki = 3200 nM T72458 CUW4Y6 44434778 Ki = 3400 nM T72458 CH8WT0 44434780 Ki = 12000 nM T72458 CL9K2D 44434781 Ki = 2600 nM T72458 CJ12GC 44434782 Ki = 9200 nM T72458 CFBX46 44434785 Ki = 7800 nM T72458 C0KB8P 44434787 Ki = 7400 nM T72458 C0M2VI 44434790 Ki = 179000 nM T72458 CH3UV8 44434794 Ki = 149000 nM T72458 C10VDG 44434797 Ki = 179000 nM T72458 CWN02S 44434799 Ki = 150000 nM T72458 C0X1MK 44434821 Ki = 6000 nM T72458 CU1ON8 44434828 Ki = 182000 nM T72458 CBHU73 44434839 Ki = 116000 nM T72458 C20UIF 44434841 Ki = 96000 nM T72458 CA7P5L 44434843 Ki = 3400 nM T72458 CBL2D7 44434845 Ki = 3400 nM T72458 CYE25C 44434847 Ki = 38000 nM T72458 CWE0J6 44434848 Ki = 7700 nM T72458 CB39YP 44434849 Ki = 33000 nM T72458 C0ZV6S 44434850 Ki = 11000 nM T72458 C4U6LJ 44434851 Ki = 7300 nM T72458 CA4M3C 44434853 Ki = 116000 nM T72458 CVGW87 44434854 Ki = 3100 nM T72458 C3G5QO 44434855 Ki = 1200 nM T72458 C2JET5 44434856 Ki = 9200 nM T72458 C2M5VB 44434857 Ki = 16000 nM T72458 CS30KD 44434858 Ki = 25000 nM T72458 C7S1OK 44434859 Ki = 11000 nM T72458 C3AVB5 44434860 Ki = 3200 nM T72458 CZQI93 44434861 Ki = 8400 nM T72458 CC0U5Y 44434862 Ki = 2500 nM T72458 CWTI58 44434863 Ki = 4400 nM T72458 CFOM13 44434864 Ki = 7300 nM T72458 CL97ID 44434865 Ki = 18000 nM T72458 CW93VX 44434867 Ki = 5300 nM T72458 CN36OD 44434868 Ki = 6500 nM T72458 CI09FJ 44434870 Ki = 2100 nM T72458 CZE48F 44434872 Ki = 5700 nM T72458 CXTV37 44434880 Ki = 3700 nM T72458 CQ45JU 44434884 Ki = 3600 nM T72458 C8POL0 44435184 Ki = 44 nM T72458 CZ8H3M 44435220 Ki = 4800 nM T72458 CPM80E 44441633 EC50 = 189 nM T72458 C7XC6E 44441634 IC50 = 1490 nM T72458 CU93IR 44441635 IC50 = 759 nM T72458 CD25AP 44441636 IC50 = 22.2 nM T72458 CQL07M 44441637 EC50 = 827 nM T72458 CIJ89K 44441638 IC50 = 173 nM T72458 CEHV41 44441639 EC50 = 196 nM T72458 C5D6YN 44441641 EC50 = 3.2 nM T72458 CP4TW0 44441642 IC50 = 6 nM T72458 CDC3R8 44441643 EC50 = 21 nM T72458 CU6ZN4 44441644 EC50 = 3.9 nM T72458 CNS4O1 44441645 EC50 = 28.7 nM T72458 CRL83D 44441646 EC50 = 111 nM T72458 C7EQ6Z 44441647 EC50 = 4.9 nM T72458 CHSV38 44441648 EC50 = 157 nM T72458 C3MIO4 44441681 EC50 = 6.5 nM T72458 CV3FT6 44441682 EC50 = 2174 nM T72458 CL93VK 44441683 EC50 = 563 nM T72458 CT3J4B 44441684 EC50 = 10 nM T72458 C3YRT9 44441685 EC50 = 546 nM T72458 CXQ3K8 44441686 EC50 = 151 nM T72458 CCS5T3 44441687 EC50 = 57.8 nM T72458 CHPU36 44441688 EC50 = 84.6 nM T72458 C9DT1C 44441689 EC50 = 1769 nM T72458 CV7BA9 44442899 Ki = 1200 nM T72458 CT3SE2 44442900 Ki = 510 nM T72458 CH8V0J 44442901 Ki = 340 nM T72458 C36JQH 44442902 Ki = 330 nM T72458 C92TFW 44442903 Ki = 310 nM T72458 C8R1KD 44442914 Ki = 300 nM T72458 CKPD40 44442931 Ki = 26 nM T72458 C6XZ1C 44442934 Ki = 38 nM T72458 CP4ZK7 44442941 Ki = 75 nM T72458 C3VJ6X 44442942 Ki = 37 nM T72458 C5PN4K 44442943 Ki = 22 nM T72458 COG72A 44442944 Ki = 130 nM T72458 CV7N5C 44442954 EC50 = 110 nM T72458 CY4E6X 44442956 EC50 = 230 nM T72458 CQ5KH1 44442958 Ki = 390 nM T72458 C7I2UT 44442965 Ki = 11 nM T72458 C45FRV 44442972 Ki = 220 nM T72458 C31FJZ 44442977 Ki = 76 nM T72458 CF6L4W 44442978 Ki = 35 nM T72458 CYMC97 44442981 Ki = 27 nM T72458 C7AD4H 44442985 Ki = 1200 nM T72458 C7Y0HL 44442989 Ki = 690 nM T72458 CYF4D6 44442990 Ki = 140 nM T72458 C6U3VA 44442992 Ki = 100 nM T72458 CUE72J 44442995 Ki = 17 nM T72458 CZ60QW 44442997 Ki = 5.5 nM T72458 C8EL0V 44442998 Ki = 29 nM T72458 C8ZU6S 44442999 Ki = 190 nM T72458 CJZ87H 44443000 Ki = 210 nM T72458 C03CKQ 44443001 Ki = 190 nM T72458 C7JY2F 44443002 Ki = 210 nM T72458 C10XIQ 44443003 Ki = 180 nM T72458 CKT6L8 44443004 Ki = 100 nM T72458 CY7H8L 44443005 Ki = 430 nM T72458 CY0GI2 44443006 Ki = 110 nM T72458 CB8R0W 44443007 Ki = 670 nM T72458 CC63OG 44443008 Ki = 200 nM T72458 CJK49H 44443009 Ki = 2200 nM T72458 C2D0OW 44443010 Ki = 3000 nM T72458 C83IEK 44443011 Ki = 3100 nM T72458 CZLT13 44443012 Ki = 4600 nM T72458 CKW85I 44443013 Ki = 3400 nM T72458 C98VGZ 44443014 Ki = 12 nM T72458 C0W5BQ 44443015 Ki = 25 nM T72458 CAU09V 44443016 Ki = 62 nM T72458 CC4RD1 44443017 Ki = 140 nM T72458 CCW51A 44443018 Ki = 110 nM T72458 C50KLT 44443019 Ki = 24 nM T72458 C7FU9B 44443020 Ki = 30 nM T72458 C47OXH 44443021 Ki = 44 nM T72458 CG7J0H 44443022 Ki = 90 nM T72458 CU5AM8 44443023 Ki = 3.6 nM T72458 CM80SQ 44443024 Ki = 130 nM T72458 C68ESY 44443025 Ki = 52 nM T72458 CZ3K8H 44443026 Ki = 29 nM T72458 C2VCS6 44443027 Ki = 65 nM T72458 CQU1O9 44443028 Ki = 32 nM T72458 CO90XC 44443029 Ki = 27 nM T72458 CGZ71H 44443030 Ki = 2.1 nM T72458 CLT7M0 44443031 Ki = 11 nM T72458 CBYR70 44443032 Ki = 16 nM T72458 CO51HP 44443033 Ki = 1.8 nM T72458 CQ68UV 44443034 Ki = 8.3 nM T72458 CO93SX 44443035 Ki = 0.5 nM T72458 C0WH1X 44443036 Ki = 110 nM T72458 C9IZ0Y 44443037 Ki = 190 nM T72458 C1GJ5L 44443038 Ki = 1800 nM T72458 CF2UI0 44443039 Ki = 2800 nM T72458 CR40SE 44443040 Ki = 1300 nM T72458 C8HOB9 44443041 Ki = 750 nM T72458 CRUJ10 44443042 Ki = 1300 nM T72458 CXI2N5 44443043 Ki = 2700 nM T72458 CM2P9T 44443044 Ki = 1500 nM T72458 C8JA5O 44444425 Ki = 520 nM T72458 CK79AB 44444427 Ki = 4800 nM T72458 C5N4FT 44444429 Ki = 1150 nM T72458 CDWO25 44444430 Ki = 1100 nM T72458 C7B9FO 44444431 Ki = 1700 nM T72458 C6DGU3 44444432 Ki = 220 nM T72458 CTD12E 44444433 Ki = 280 nM T72458 C0V8UC 44444434 Ki = 250 nM T72458 CWGI62 44444435 Ki = 580 nM T72458 C73MYX 44444436 Ki = 320 nM T72458 C2QC4X 44444437 Ki = 420 nM T72458 CHOG98 44444438 Ki = 490 nM T72458 CQ37OR 44444440 Ki = 1200 nM T72458 C02WEC 44444441 Ki = 1200 nM T72458 C92TOP 44444442 Ki = 1100 nM T72458 CDS4U1 44444443 Ki = 320 nM T72458 C6M3VD 44444444 Ki = 550 nM T72458 C9WP5E 44444445 Ki = 950 nM T72458 CUG3B4 44444446 Ki = 360 nM T72458 CL31BQ 44444447 Ki = 840 nM T72458 C0EA1Z 44444448 Ki = 92 nM T72458 CGEZ90 44444449 Ki = 510 nM T72458 C98HTN 44444450 Ki = 230 nM T72458 CFN72H 44444452 Ki = 270 nM T72458 CT69RO 44444454 Ki = 520 nM T72458 CU24DB 44444457 Ki = 240 nM T72458 CYO9U6 44444460 Ki = 190 nM T72458 CL6TV9 44444462 Ki = 1600 nM T72458 CPJI69 44444465 Ki = 1400 nM T72458 C60GBK 44444468 Ki = 450 nM T72458 CQCK08 44444483 Ki = 13 nM T72458 C4ZDW3 44444490 Ki = 47 nM T72458 CB39DL 44444493 Ki = 7.1 nM T72458 CE5CR4 44444495 Ki = 4.7 nM T72458 CBO36Z 44444497 Ki = 11 nM T72458 CIOT60 44444499 Ki = 4.4 nM T72458 C5DWM0 44444500 EC50 = 6.9 nM T72458 C3VL8P 44444502 Ki = 8.9 nM T72458 CD7N9T 44444504 Ki = 7.7 nM T72458 CL17PU 44444505 Ki = 17.3 nM T72458 CDWM65 44444507 Ki = 4.9 nM T72458 C3PST9 44444508 Ki = 47 nM T72458 CIE0P1 44444509 Ki = 10 nM T72458 COS36P 44444510 EC50 = 6.6 nM T72458 C2YX7D 44444511 Ki = 87 nM T72458 CXT65M 44447207 Ki = 810 nM T72458 C7X9AU 44447208 Ki = 280 nM T72458 CVS9K1 44447209 Ki = 130 nM T72458 CY19GE 44447210 Ki = 170 nM T72458 CL03RO 44447211 Ki = 130 nM T72458 CVR68Z 44447212 Ki = 250 nM T72458 COI65T 44447214 Ki = 120 nM T72458 C9PYC4 44447218 Ki = 230 nM T72458 CNJ3I2 44447221 Ki = 38 nM T72458 C9JN4F 44447222 Ki = 170 nM T72458 C4HB7O 44447223 Ki = 190 nM T72458 CT6R7Z 44447224 Ki = 100 nM T72458 CEF6Y1 44447225 Ki = 180 nM T72458 CEK98D 44447226 Ki = 280 nM T72458 CDYL03 44447227 Ki = 71 nM T72458 CW27UZ 44447228 Ki = 260 nM T72458 C8GJI0 44447229 Ki = 290 nM T72458 CY2E8N 44447230 Ki = 180 nM T72458 C3MB7S 44447231 Ki = 330 nM T72458 CS2P5V 44447232 Ki = 200 nM T72458 C8DTJ1 44447233 Ki = 280 nM T72458 CV85GR 44447234 Ki = 74 nM T72458 CG02YX 44447235 Ki = 87 nM T72458 C4APF9 44447236 Ki = 110 nM T72458 CG3W0E 44447237 Ki = 380 nM T72458 CM68RP 44447238 Ki = 37 nM T72458 C60TVF 44447239 Ki = 790 nM T72458 CJ6ZW7 44447240 Ki = 40 nM T72458 CN2X1M 44447241 Ki = 30 nM T72458 CLHT47 44447242 Ki = 28 nM T72458 CYGJ75 44447243 Ki = 410 nM T72458 C9VME8 44447244 Ki = 590 nM T72458 CIS36F 44447245 Ki = 120 nM T72458 CAD46C 44447246 Ki = 1100 nM T72458 CG0L1J 44447247 Ki = 2100 nM T72458 C73SEZ 44447248 Ki = 480 nM T72458 CHO8Y4 44447249 Ki = 43 nM T72458 CG3FA6 44447250 Ki = 10 nM T72458 C0WQO6 44447251 EC50 = 2 nM T72458 C2F7YZ 44447764 Ki = 550 nM T72458 C8MK6X 44447765 Ki = 340 nM T72458 C8Q7FC 44447767 Ki = 98 nM T72458 C8OG4F 44447768 Ki = 96 nM T72458 CE1G2K 44447769 Ki = 190 nM T72458 CM8F0V 44447770 Ki = 110 nM T72458 CS80GC 44447771 Ki = 560 nM T72458 CWN9X8 44447772 Ki = 56 nM T72458 C4A7BL 44447773 Ki = 52 nM T72458 C9MVL5 44447774 Ki = 160 nM T72458 CPL5B2 44447776 Ki = 110 nM T72458 CQ8BE5 44447777 Ki = 11 nM T72458 C6V5UQ 44447778 Ki = 120 nM T72458 C9NXS5 44447779 Ki = 7.2 nM T72458 C8YZ0G 44447780 Ki = 17 nM T72458 CAK75F 44447781 Ki = 53 nM T72458 CVUW60 44447785 Ki = 11 nM T72458 C86ATQ 44447787 Ki = 130 nM T72458 C3V9UN 44447791 Ki = 12 nM T72458 C9O7VQ 44447801 Ki = 94 nM T72458 CU7S8G 44447802 Ki = 74 nM T72458 C5SY1J 44447803 Ki = 18 nM T72458 CCRY28 44447804 Ki = 6.5 nM T72458 CWDG08 44447805 Ki = 190 nM T72458 C0C7VJ 44447806 Ki = 40 nM T72458 C7QT3I 44447807 Ki = 45 nM T72458 C6KPH5 44447808 Ki = 97 nM T72458 CQLZ83 44447809 Ki = 330 nM T72458 C9KNO3 44447810 Ki = 54 nM T72458 C4X7YK 44447811 Ki = 1800 nM T72458 C3L4FZ 44447812 Ki = 78 nM T72458 C4OWP8 44447816 Ki = 180 nM T72458 C5MF9J 44447817 Ki = 79 nM T72458 CFL6R4 44447818 Ki = 92 nM T72458 CXAF32 44447819 Ki = 62 nM T72458 C37AZY 44447820 Ki = 52 nM T72458 C9OBG6 44447821 Ki = 55 nM T72458 CB3KW6 44447822 Ki = 59 nM T72458 CDX4V1 44447823 Ki = 42 nM T72458 CB1GF4 44447824 Ki = 68 nM T72458 C14OSV 44447847 IC50 = 2400 nM T72458 C03AQC 44447849 IC50 = 1500 nM T72458 CR1M0J 44447851 IC50 = 960 nM T72458 CRI7M8 44448436 IC50 = 127.6 nM T72458 C6I4PC 44448477 IC50 = 101.1 nM T72458 C08BMY 44448479 EC50 = 120.5 nM T72458 C2FA5H 44448480 EC50 = 1922 nM T72458 CWB1I0 44448515 IC50 = 28.1 nM T72458 CP35SZ 44448554 IC50 = 22.7 nM T72458 C8TK3Y 44448588 IC50 = 9.8 nM T72458 C0C7KI 44448590 EC50 = 4.6 nM T72458 CMYO10 44448628 IC50 = 37.2 nM T72458 CQHR95 44448629 EC50 = 2.1 nM T72458 C78XDT 44448631 EC50 = 13.4 nM T72458 C8H1UT 44448660 EC50 = 2.8 nM T72458 CCV7B1 44448661 EC50 = 110.8 nM T72458 CL28KE 44448677 IC50 = 82.2 nM T72458 CGZ1F9 44448698 EC50 = 155.6 nM T72458 CYAN15 44449216 EC50 = 565 nM T72458 CTP3D6 44453826 Ki > 100000 nM T72458 C4FV3C 44453850 Ki > 25000 nM T72458 CEI35V 44453902 Ki = 6700 nM T72458 CUPG04 44453903 EC50 > 25000 nM T72458 CBV08D 44455891 Ki = 290 nM T72458 C9L0JY 44455892 Ki = 260 nM T72458 CH1DK5 44455893 Ki = 51 nM T72458 C9GLW5 44455922 Ki = 7.5 nM T72458 CW2PJ8 44455923 Ki = 2050 nM T72458 CAK1U0 44455956 Ki = 470 nM T72458 CF3W1O 44455957 Ki = 560 nM T72458 C92TBV 44455958 Ki = 61 nM T72458 CSVD47 44455996 Ki = 370 nM T72458 CN89EI 44455997 Ki = 3700 nM T72458 CP2EH4 44456027 Ki = 5.3 nM T72458 CH5BY0 44456102 Ki = 1 nM T72458 CI1PL0 44456137 Ki = 2.1 nM T72458 CCW1A3 44456138 Ki = 7.3 nM T72458 CE9VC8 44456183 Ki = 2.2 nM T72458 CD8EJ4 44456184 Ki = 2 nM T72458 C63APB 44456219 Ki = 4.7 nM T72458 CE0P7K 44456222 Ki = 1 nM T72458 CF40UY 44456259 Ki = 5.3 nM T72458 CFD8Z5 44456304 Ki = 4.6 nM T72458 CFD62Q 44456336 Ki = 7.6 nM T72458 C8N0CX 44456368 Ki = 90 nM T72458 CM69AH 44456410 Ki = 7.2 nM T72458 CGLM70 44456416 Ki = 850 nM T72458 C6GL4V 44456460 Ki = 7800 nM T72458 CU7JV8 44456461 Ki = 250 nM T72458 CC64AO 44457043 IC50 = 100 nM T72458 CZ36WX 44457067 IC50 = 60 nM T72458 C4DL5C 44469677 IC50 > 10000 nM T72458 CA5MU1 44562283 Ki = 1700 nM T72458 C27VXC 44562284 Ki = 5800 nM T72458 CA1GN0 44562285 Ki > 10000 nM T72458 C7Z4UN 44562286 Ki = 13 nM T72458 C5CIX6 44562287 Ki = 9.4 nM T72458 C4PR2V 44562288 Ki = 18 nM T72458 C8QL9K 44562289 Ki = 65 nM T72458 C4JKU5 44562323 Ki > 10000 nM T72458 CNF96U 44562324 Ki = 38 nM T72458 COB0Q8 44562361 Ki = 110 nM T72458 C8VGJ4 44562362 Ki = 380 nM T72458 C7B3HD 44562363 Ki = 330 nM T72458 C6JX0A 44562364 Ki = 89 nM T72458 C02QLT 44562365 Ki = 1400 nM T72458 CF5W2K 44562366 Ki = 42 nM T72458 CLFX67 44562367 Ki = 390 nM T72458 CAF74R 44562368 Ki = 110 nM T72458 CHN87Y 44562389 Ki = 3200 nM T72458 C1ZH5L 44562390 Ki > 10000 nM T72458 CA6ZN2 44562391 Ki = 53 nM T72458 CQ8Z5M 44562392 Ki = 83 nM T72458 CKB04G 44562398 Ki = 21 nM T72458 CEQ6Y1 44562399 Ki = 15 nM T72458 C18SIO 44562400 Ki = 120 nM T72458 CSC76I 44562401 Ki = 350 nM T72458 C0SD6C 44562402 Ki = 2 nM T72458 C21YKQ 44562412 Ki = 350 nM T72458 CL6ZR3 44562413 Ki = 1200 nM T72458 CU92FG 44562414 Ki = 24 nM T72458 C93SKQ 44562421 Ki = 33 nM T72458 CA53WV 44562422 Ki = 31 nM T72458 CN3Y7I 44562423 Ki = 26 nM T72458 C5F3XU 44562424 Ki = 110 nM T72458 C9SVX4 44562438 Ki = 91 nM T72458 CCIS23 44562439 Ki = 13 nM T72458 CPSC21 44562440 Ki = 8.3 nM T72458 CTN82A 44562457 Ki = 16 nM T72458 CSVX92 44562458 Ki = 46 nM T72458 CU98AG 44562459 Ki = 21 nM T72458 CQ0I1K 44562460 Ki = 3.2 nM T72458 CY14WQ 44562475 Ki = 2 nM T72458 CQV9B7 44562476 Ki = 1.7 nM T72458 C0VXR6 44562477 Ki = 4.2 nM T72458 C8EQD4 44562478 Ki = 7.7 nM T72458 CAM86F 44562495 Ki = 4.7 nM T72458 CAG1U4 44562496 Ki = 870 nM T72458 C4XFR3 44562497 Ki = 26 nM T72458 CRQW35 44562498 Ki = 110 nM T72458 C7V4WX 44562518 Ki = 29 nM T72458 CXDB43 44562519 Ki = 47 nM T72458 CP98CO 44562520 Ki = 54 nM T72458 CB18VE 44562538 Ki = 66 nM T72458 C8RQE4 44562539 Ki = 66 nM T72458 CF9N1W 44562540 Ki = 32 nM T72458 C94MEZ 44562541 Ki = 23 nM T72458 C0L6BJ 44562558 Ki = 11 nM T72458 CH42ZU 44562559 Ki = 11 nM T72458 CQ3J2B 44562560 Ki = 280 nM T72458 C2L6FI 44562561 Ki = 9 nM T72458 CV79ML 44562593 Ki > 10000 nM T72458 C1WU4Q 44562594 Ki = 560 nM T72458 C0GTB1 44562595 Ki = 230 nM T72458 C5OJ6B 44562596 Ki = 150 nM T72458 CK5WI0 44562597 Ki = 28 nM T72458 C3NSL9 44562598 Ki = 49 nM T72458 C6ILB9 44562599 Ki = 26 nM T72458 CQ8J9K 44569175 EC50 = 2 nM T72458 CL8GU3 44569176 EC50 = 0.9 nM T72458 C97DSW 44577054 Ki = 83 nM T72458 C2FP9E 44577055 Ki = 210 nM T72458 CP56CV 44577056 Ki = 180 nM T72458 C4WP0Z 44577059 Ki = 5.3 nM T72458 CD3T1I 44577060 Ki = 7.5 nM T72458 CQ1M9C 44577061 Ki = 3.1 nM T72458 C6FI8E 44577062 Ki = 4.1 nM T72458 CJ6GZ3 44577063 Ki = 5.4 nM T72458 CHJ6Z1 44577064 Ki = 24 nM T72458 CY4QE9 44577087 Ki = 26 nM T72458 CGF37X 44577088 Ki = 27 nM T72458 CR6Q2S 44577089 Ki = 23 nM T72458 CWOK70 44577090 Ki = 10 nM T72458 C4FSH3 44577091 Ki = 3.4 nM T72458 CF8PL1 44577092 Ki = 1.1 nM T72458 CM6X5S 44577093 Ki = 0.8 nM T72458 CGTV08 44577094 Ki = 3.3 nM T72458 C0YI4V 44577095 Ki = 1.3 nM T72458 CEJ96P 44577510 EC50 = 37 nM T72458 C6Y1BS 44577515 IC50 > 5000 nM T72458 C8B1WR 44577520 IC50 > 1000 nM T72458 C3NSW7 44577523 IC50 > 1000 nM T72458 CR5ZS2 44583562 EC50 = 11 nM T72458 CWFB17 44583567 IC50 = 1.2 nM T72458 CO7X1P 45277088 Ki < 10000 nM T72458 C26EWX 45277089 Ki < 10000 nM T72458 C6X4ER 45277090 Ki < 10000 nM T72458 CH7I1J 45277245 Ki < 10000 nM T72458 CHWX12 46202887 EC50 > 10000 nM T72458 CXM2I4 46202891 EC50 = 53 nM T72458 CM68TW 46202892 EC50 = 108 nM T72458 CCE2L7 46203212 EC50 = 644 nM T72458 C02XLV 46203213 EC50 = 3630 nM T72458 C4N2CP 46203214 EC50 = 11100 nM T72458 CJB6H0 46203215 Ki = 107 nM T72458 CKA84X 46203216 EC50 = 147 nM T72458 CO8H3A 46203515 EC50 = 51 nM T72458 CO95IX 46203516 EC50 = 69 nM T72458 CVW98L 46203517 EC50 = 40 nM T72458 CY12SB 46228659 EC50 > 30000 nM T72458 C10VXP 46228660 EC50 = 338.84 nM T72458 C8XUS4 46228689 EC50 = 794.33 nM T72458 C5FVJ9 46228690 EC50 = 100 nM T72458 CCK7I1 46228725 EC50 > 30000 nM T72458 CD5Q8V 46228726 EC50 = 1071.52 nM T72458 CJ7R0X 46228763 EC50 > 30000 nM T72458 CYD2R3 46228764 EC50 = 1258.93 nM T72458 CQ53EA 46228813 EC50 = 2884.03 nM T72458 CMX28H 46228814 EC50 = 1047.13 nM T72458 C7FAY5 46228815 EC50 = 660.69 nM T72458 C82NVP 46228841 EC50 > 30000 nM T72458 CEDL84 46228842 EC50 > 30000 nM T72458 CP86QH 46228843 EC50 > 30000 nM T72458 C4BD8Z 46228844 EC50 > 30000 nM T72458 CR6PF0 46228845 EC50 > 30000 nM T72458 CCN14H 46228846 EC50 = 165.96 nM T72458 C3T1NY 46228847 EC50 > 30000 nM T72458 COW85F 46228848 EC50 > 30000 nM T72458 CZLY24 46228849 EC50 > 30000 nM T72458 C5VAN7 46228850 EC50 > 30000 nM T72458 C0X9KS 46228888 EC50 > 30000 nM T72458 CDE7N9 46865980 EC50 = 3900 nM T72458 CBI76Q 46884747 IC50 = 89 nM T72458 CQ28TZ 46884748 EC50 = 37.2 nM T72458 CD3E4C 46885323 Ki = 264 nM T72458 CNH0I9 46885324 EC50 = 255 nM T72458 C53CEM 46885325 EC50 = 159 nM T72458 CPKC94 46885326 EC50 = 288 nM T72458 C65EKV 46885366 EC50 = 19 nM T72458 CNW43Y 46885367 EC50 = 55 nM T72458 CE4SF8 46885368 EC50 = 105 nM T72458 C4YX1U 46885369 EC50 = 73 nM T72458 CLY30Q 46885414 EC50 = 81 nM T72458 CV23JL 46885415 EC50 = 32 nM T72458 C7M3HS 46885416 EC50 = 374 nM T72458 CHPS01 46885417 EC50 = 18 nM T72458 C4SVE1 46885480 EC50 = 15 nM T72458 C5QI7J 46885481 EC50 = 5 nM T72458 COU5X2 46885482 EC50 = 6 nM T72458 CU28GA 46885483 EC50 = 4 nM T72458 CG9NJ1 46885523 EC50 = 7 nM T72458 CS90MN 46885524 EC50 = 21 nM T72458 CWI08O 46885525 EC50 = 89 nM T72458 CQ94VM 46885526 EC50 = 82 nM T72458 C90ABZ 46885558 EC50 = 4 nM T72458 C0U7TG 46885559 EC50 = 117 nM T72458 C0MI3C 46885560 EC50 = 243 nM T72458 C50BUQ 46885561 EC50 = 111 nM T72458 CL86JU 46885621 EC50 = 15 nM T72458 CFJ0C1 46885622 EC50 = 220 nM T72458 CX4K9T 46885674 EC50 = 1116 nM T72458 C0Y9NF 46885711 EC50 = 30 nM T72458 C3O5BR 46885712 EC50 = 18 nM T72458 CA82IZ 46885713 EC50 = 347 nM T72458 CG6XN0 46885759 EC50 = 6 nM T72458 CK8D6G 46885760 EC50 = 45 nM T72458 C0C8GN 46885761 EC50 = 62 nM T72458 CY30PG 46885815 EC50 = 46 nM T72458 CEA70O 46885816 EC50 = 126 nM T72458 C6ZUB5 46885817 EC50 = 626 nM T72458 C8LHF6 46885861 EC50 = 962 nM T72458 CAZN09 46885862 EC50 = 130 nM T72458 CWN89S 46885863 Ki = 346 nM T72458 CKQ4X2 46885906 EC50 = 85 nM T72458 C8UTI7 46885907 EC50 = 61 nM T72458 CFC5L1 46885972 EC50 = 69 nM T72458 CUDE25 46885973 EC50 = 91 nM T72458 C3FN1Z 46885974 EC50 = 52 nM T72458 CDH7N3 46886010 EC50 = 257 nM T72458 CO3S1Q 46905544 Ki = 31392 nM T72458 C96XEU 46905545 Ki = 4756 nM T72458 CDY4U0 46911588 EC50 = 2.1 nM T72458 C29LQB 46919520 EC50 = 2.7 nM T72458 CK41RF 46930942 Ki = 1300 nM T72458 CIGV98 46930943 Ki = 350 nM T72458 C8Y2QS 49798104 IC50 = 398.11 nM T72458 C6LEM8 49798106 IC50 = 31.62 nM T72458 C8EG6Y 49798111 IC50 = 1258.93 nM T72458 C24DUW 49798112 IC50 = 251.19 nM T72458 CQS6G8 49798149 IC50 = 200 nM T72458 C1EMQ2 49861348 EC50 = 12 nM T72458 C9QU3G 49862375 EC50 = 5.4 nM T72458 C4WHG2 49862376 EC50 = 10 nM T72458 CPZI97 49862377 EC50 = 6.4 nM T72458 CY7R2T 49862378 EC50 = 9.7 nM T72458 C7GA4I 49862425 EC50 = 19 nM T72458 C1BC2M 49862426 IC50 = 150 nM T72458 C2ZHD1 49862478 EC50 = 19 nM T72458 CN1AJ5 49862662 IC50 = 31.4 nM T72458 CT69NY 49862663 IC50 = 479.2 nM T72458 CW2KQ0 49862664 EC50 = 78.1 nM T72458 C1X3WL 49862665 EC50 = 2.6 nM T72458 CG78ZY 49862736 EC50 = 1.1 nM T72458 C8GVY6 49862737 IC50 = 52.5 nM T72458 C0N8IJ 49862738 IC50 = 6.6 nM T72458 C5MZ9X 49862739 IC50 = 11.9 nM T72458 CBIK17 49862740 IC50 = 44.3 nM T72458 CHX09I 49862741 IC50 = 7.6 nM T72458 CZVN53 49862742 EC50 = 17.1 nM T72458 C8M2TH 49862743 EC50 = 7.4 nM T72458 C9T8SI 49862744 IC50 = 150.7 nM T72458 C8XA3E 49862745 EC50 = 1.5 nM T72458 CEX17U 49862746 IC50 = 3.6 nM T72458 CA2RN4 49862747 IC50 = 2.3 nM T72458 CD5ZR4 49862748 EC50 = 0.6 nM T72458 CPVE31 49862749 EC50 = 3.1 nM T72458 CNY2L7 49862750 EC50 = 0.8 nM T72458 CV6YZ5 49862751 EC50 = 2.9 nM T72458 CFR38H 50899078 EC50 = 0.23 nM T72458 C0QD9I 51346770 Ki = 392 nM T72458 C30PGL 51346771 Ki = 403 nM T72458 CBQN64 52918026 EC50 = 22 nM T72458 CZ8P7W 52940633 EC50 = 14 nM T72458 CZG5F1 52941830 EC50 = 2.4 nM T72458 C5RGD8 52943036 EC50 = 1000 nM T72458 C3XP8F 52943061 IC50 = 1.3 nM T72458 CB71IN 52944242 EC50 = 4.2 nM T72458 CDZ3L2 52945472 IC50 = 1.9 nM T72458 CQN8V6 52947911 IC50 = 9.7 nM T72458 CG5TJ0 53240339 IC50 = 515 nM T72458 CQ7O3U 54584301 IC50 = 16 nM T72458 C8PIL3 54584302 EC50 = 58 nM T72458 CN6F2C 54586246 IC50 = 5.1 nM T72458 CEU0M6 54587278 IC50 = 0.78 nM T72458 CLB28F 56595060 Ki = 330 nM T72458 CF34IC 56659456 EC50 = 0.25 nM T72458 CM94BT 56659465 EC50 = 53 nM T72458 C8BF3M 56659466 EC50 = 0.91 nM T72458 C5V2RD 56659467 EC50 = 1.3 nM T72458 CN41CZ 56659468 EC50 = 4.3 nM T72458 CF3LR1 56662904 EC50 = 0.69 nM T72458 C27DXA 56662925 EC50 = 1.4 nM T72458 CNSK26 56662927 EC50 = 1.9 nM T72458 C8C9IS 56666386 EC50 = 0.37 nM T72458 C3OM7E 56666397 EC50 = 32 nM T72458 CYKJ48 56669816 EC50 = 28 nM T72458 CPT38A 56669817 IC50 = 12 nM T72458 CFU39L 56669819 EC50 = 0.59 nM T72458 CCLJ91 56669820 EC50 = 0.76 nM T72458 C8H9RM 56672278 IC50 = 4900 nM T72458 C2YB1Q 56673302 IC50 = 0.71 nM T72458 C69KAM 56673304 EC50 = 9.9 nM T72458 C1GI2N 56673305 EC50 = 1.1 nM T72458 CE7CI0 56676614 EC50 = 1.2 nM T72458 CJDZ96 56676631 IC50 = 2.5 nM T72458 C7VO5D 56676632 EC50 = 0.8 nM T72458 CJZ5V3 56676633 IC50 = 6.6 nM T72458 CYQ3A6 56676634 EC50 = 307 nM T72458 CA1Q8I 56676635 EC50 = 2.3 nM T72458 C9V7LA 56676638 EC50 = 0.38 nM T72458 CEA19V 56676639 EC50 = 1.1 nM T72458 CLB0G3 56679956 EC50 = 3.8 nM T72458 C47TEG 56679964 EC50 = 12 nM T72458 CAYG58 56679968 EC50 = 1 nM T72458 CP7UR2 56683296 EC50 = 2.9 nM T72458 C9VT6Z 56683297 EC50 = 4.2 nM T72458 CFBT37 56683299 EC50 = 1.6 nM T72458 CZ7WN1 56683300 EC50 = 1.7 nM T72458 CB96KR 56683301 EC50 = 0.98 nM T72458 CTSB57 56850936 Ki = 988 nM T72458 C1U2DB 56851057 Ki = 254 nM T72458 C2WAO4 57634921 EC50 = 2 nM T72458 C4VT5C 57634925 EC50 = 0.47 nM T72458 CKW2T0 57646411 EC50 = 0.04 nM T72458 C8F5XG 57646441 Ki = 0.12 nM T72458 CS2E3H 58658553 EC50 = 6.2 nM T72458 CH1LU3 58777892 Ki = 70 nM T72458 C5P1EC 58777970 Ki = 190 nM T72458 CBM78A 59077913 EC50 = 44 nM T72458 CD1C7S 60168008 Ki = 70 nM T72458 CP6V2L 70681741 Ki = 1800 nM T72458 CPJ3U7 70681742 Ki = 380 nM T72458 C3PS2N 70681743 Ki = 160 nM T72458 CS27GN 70682904 Ki = 36000 nM T72458 C73SKU 70682946 EC50 = 29 nM T72458 CBY2K9 70683600 IC50 = 29 nM T72458 C06RGO 70683847 Ki = 5500 nM T72458 C65FDK 70683848 Ki = 1000 nM T72458 C0O6QG 70685712 IC50 = 20 nM T72458 CCU8P0 70685980 Ki = 900 nM T72458 CAJ5U0 70685981 Ki = 1000 nM T72458 CP7J6R 70688108 Ki = 5500 nM T72458 C3O4SK 70688109 Ki = 6600 nM T72458 CEFQ39 70688110 Ki = 670 nM T72458 CNH4F5 70688111 Ki = 400 nM T72458 CPJ08L 70688853 Ki = 0.33 nM T72458 CU86WQ 70689887 IC50 = 24 nM T72458 CB2X0A 70689888 IC50 = 17 nM T72458 CMKH31 70690145 Ki = 5000 nM T72458 C63ULO 70690146 Ki = 5800 nM T72458 CPM3N9 70690147 Ki = 2600 nM T72458 C2T3GP 70690148 Ki = 6200 nM T72458 C81JGS 70692049 IC50 = 40 nM T72458 C2P3IN 70692050 EC50 = 18 nM T72458 COSQ85 70694364 Ki = 5300 nM T72458 C3G7MZ 70695694 EC50 = 110 nM T72458 C97FOR 70696210 IC50 = 25 nM T72458 C2O7TA 71449047 EC50 = 6.1 nM T72458 CH0F4A 71449048 EC50 > 10000 nM T72458 C1JN2M 71449119 EC50 = 13 nM T72458 CMS5R6 71449140 Ki = 166000 nM T72458 CJPX32 71449204 EC50 = 52 nM T72458 C93FSV 71450911 Ki = 89 nM T72458 C8IXY4 71450912 Ki = 150 nM T72458 CK43RW 71450919 Ki = 500 nM T72458 C6BK5F 71450920 Ki = 3900 nM T72458 CBP20G 71452716 EC50 = 25 nM T72458 CKCN10 71452720 IC50 = 16 nM T72458 C8JMR2 71452721 Ki = 49 nM T72458 C2AGS1 71452731 Ki = 950 nM T72458 CEB0P9 71452732 Ki = 2500 nM T72458 CNPI97 71452733 Ki = 700 nM T72458 CICH01 71452734 Ki = 410 nM T72458 CD94NF 71452735 Ki = 230 nM T72458 CV0J8X 71452824 IC50 = 20 nM T72458 CN4EJ2 71452825 IC50 = 8 nM T72458 CW8OE1 71452826 IC50 = 30 nM T72458 C50LPK 71454491 EC50 = 12 nM T72458 CV4ZM6 71454492 EC50 = 49 nM T72458 C3D7ZL 71454495 Ki = 78 nM T72458 COP19B 71454508 Ki = 150 nM T72458 CN58TM 71454509 Ki = 170 nM T72458 CNB53G 71454510 Ki = 50 nM T72458 CY16AM 71454518 Ki = 15000 nM T72458 CPX03G 71456219 IC50 = 3700 nM T72458 C07WXP 71456220 EC50 > 10000 nM T72458 CQPB08 71456236 EC50 = 16 nM T72458 C05GFW 71456243 Ki = 53 nM T72458 CNRV69 71456245 IC50 = 18 nM T72458 C3NS6M 71456246 EC50 = 740 nM T72458 C3E1NT 71456250 Ki = 1600 nM T72458 C5VH2T 71456251 Ki = 280 nM T72458 CA5GY9 71458041 EC50 = 8 nM T72458 CQZ48M 71458046 Ki = 240 nM T72458 CU17GR 71458055 Ki = 7700 nM T72458 C93UJT 71458056 Ki = 4800 nM T72458 C6WOE4 71458057 Ki = 240 nM T72458 CG89OM 71458058 Ki = 140 nM T72458 C1WR2D 71458059 Ki = 80 nM T72458 C6YR0U 71458117 IC50 > 10000 nM T72458 C3V0DA 71459896 EC50 = 45 nM T72458 CO8C4B 71459937 IC50 = 280 nM T72458 CJ52CU 71459938 IC50 = 22 nM T72458 CS9Y6R 71459941 Ki = 530 nM T72458 CCRG02 71459942 Ki = 180 nM T72458 CU2A1J 71461601 EC50 = 570 nM T72458 CUJS47 71461649 EC50 = 8.6 nM T72458 C3HLD7 71461652 IC50 = 560 nM T72458 C5J2CA 71461656 Ki = 2100 nM T72458 CECQ16 71461657 Ki = 4200 nM T72458 C24GWM 71461662 Ki = 70000 nM T72458 CZ94CM 71461730 IC50 = 0.89 nM T72458 C9E2DM 71717586 IC50 = 4900 nM T72458 CYA8G1 71717886 EC50 = 26 nM T72458 CPH79G 71769787 Ki = 1.8 nM T72458 CMH31J 71769905 Ki = 600 nM T72458 C8KS6E 71770031 Ki = 2.4 nM T72458 CWH6T3 72548703 IC50 = 0.21 nM T72458 CV8K5U 73345513 Ki = 4800 nM T72458 C4IAM6 73345514 Ki = 4.6 nM T72458 CG3H2F 73345549 IC50 = 30 nM T72458 C1A5SK 73345616 IC50 = 74 nM T72458 CI0DV9 73345617 IC50 > 5000 nM T72458 C62DYB 73345878 IC50 = 40 nM T72458 CYMH60 73347015 Ki = 1.5 nM T72458 C31UAJ 73347130 EC50 = 8 nM T72458 C7DYR4 73347133 EC50 = 2 nM T72458 CZ91TE 73347138 IC50 = 570 nM T72458 CK46SP 73347139 IC50 = 4700 nM T72458 CX9LF8 73347140 IC50 = 990 nM T72458 CU1T4A 73347614 Ki = 6 nM T72458 CW8F4U 73348170 EC50 = 0.3 nM T72458 C4SR8Z 73348617 EC50 = 3.3 nM T72458 CK69FV 73348634 EC50 = 3 nM T72458 C6VK5T 73350013 IC50 = 620 nM T72458 CS4I5R 73350057 Ki = 1.01 nM T72458 CI9FS8 73350149 EC50 = 65 nM T72458 CI07CR 73350214 EC50 = 5 nM T72458 CMLR03 73350220 IC50 = 160 nM T72458 CPW67D 73350705 Ki = 0.14 nM T72458 C3EF0P 73351617 Ki = 0.22 nM T72458 CCF87P 73351717 EC50 = 25 nM T72458 CKWH98 73351727 IC50 = 720 nM T72458 CWHE24 73351850 EC50 = 140 nM T72458 C1L7HK 73353100 Ki = 5.7 nM T72458 CJL0D3 73353101 EC50 = 53 nM T72458 CR9N5P 73353187 EC50 = 3162.28 nM T72458 C8C0LW 73353205 IC50 = 4700 nM T72458 CGVC68 73353206 IC50 = 1600 nM T72458 CV27XE 73353216 EC50 = 290 nM T72458 CK2X0G 73353271 IC50 = 3.5 nM T72458 CS3FZ1 73353454 IC50 = 12 nM T72458 CK23FW 73354573 Ki = 2.2 nM T72458 CIEJ89 73354618 Ki = 1.5 nM T72458 CA4MR1 73354641 IC50 = 4 nM T72458 CXZD68 73354698 EC50 = 1995.26 nM T72458 C15BNT 73354704 EC50 = 65 nM T72458 C0ISQ4 73354708 IC50 = 1000 nM T72458 CJS25D 73354709 IC50 > 10000 nM T72458 C7OL2D 73354716 EC50 = 45 nM T72458 C7OT4D 73354780 EC50 = 0.11 nM T72458 CA8MQ1 73354785 IC50 = 230 nM T72458 CB6G1I 73355183 Ki = 150 nM T72458 CAWT96 73355184 Ki = 37 nM T72458 C17PEL 73356313 IC50 = 3.7 nM T72458 CT5UP1 73356732 Ki = 1.7 nM T72458 CR8M0O 73356733 Ki = 1.5 nM T72458 CA4U8O 90643802 EC50 = 0.24 nM T72458 CGBM80 90643803 EC50 = 0.12 nM T72458 CMAX81 90643804 EC50 = 0.26 nM T72458 CI05XM 90643805 EC50 = 0.29 nM T72458 CUJR85 90643806 EC50 = 0.4 nM T72458 C5N1DE 90643807 EC50 = 0.45 nM T72458 C1K0SJ 90643808 EC50 = 0.21 nM T72458 CSL28O 90643809 EC50 = 0.19 nM T72458 C4K7OV 90643810 EC50 = 1.06 nM T72458 CI50KM 90643811 EC50 = 40 nM T72458 CNE2F6 90643812 EC50 = 75 nM T72458 C36YQG 90643813 EC50 = 17 nM T72458 CS03VB 90643814 EC50 = 46 nM T72458 C68MKS 90643815 EC50 = 15 nM T72458 CJZ4V6 90643816 EC50 = 48 nM T72458 CHWK42 90643817 EC50 = 76 nM T72458 C9RH7W 90643818 EC50 = 1.9 nM T72458 CTN29R 90643819 EC50 = 204 nM T72458 CWL31Q 90643820 EC50 > 10000 nM T72458 CY70XF 90643821 EC50 = 5.3 nM T72458 CHV9I8 90643822 EC50 = 195 nM T72458 CAI8R0 90643823 EC50 = 28 nM T72458 CZ07JO 90643824 EC50 = 5.1 nM T72458 CRE52K 90643825 EC50 = 114 nM T72458 C36QSP 90643826 EC50 = 20 nM T72458 COES74 90643827 EC50 = 4.26 nM T72458 C83TIZ 90643828 EC50 = 280 nM T72458 CT7B4I 90643829 EC50 = 7.42 nM T72458 C2S5YA 90643830 EC50 = 24 nM T72458 CWDZ15 90643831 EC50 = 3.6 nM T72458 CD5C0I 90643832 EC50 = 89 nM T72458 CPX3G4 90643833 EC50 = 203 nM T72458 CM0JB7 90643834 EC50 = 2260 nM T72458 CC3T0S 90643835 EC50 = 6.65 nM T72458 C7IB3W 90643836 EC50 = 57 nM T72458 CVK16Q 90643837 EC50 = 9.6 nM T72458 CI64FK 90643838 EC50 = 120 nM T72458 CTU2B7 90643839 EC50 = 640 nM T72458 CKG73H 90643840 EC50 = 40 nM T72458 CM76IZ 90643841 EC50 = 2.6 nM T72458 C2OYM0 90643842 EC50 = 960 nM T72458 C38ZOR 90643843 EC50 = 15 nM T72458 C0K8EC 90643844 EC50 = 160 nM T72458 C8YK4D 90643845 EC50 = 15 nM T72458 CZ7W6Y 90643846 EC50 = 110 nM T72458 C5QDW8 90643847 EC50 = 22 nM T72458 CE2T4B 90643848 EC50 = 250 nM T72458 CKQ84G 90643849 EC50 = 21 nM T72458 CK58AT 90643850 EC50 = 110 nM T72458 CKP10U 90664284 IC50 = 6500 nM T72458 CP1S3T 90664642 EC50 = 82 nM T72458 CR7OX0 90664763 EC50 = 29 nM T72458 CVQ3P5 91971097 IC50 = 3300 nM T72458 C6L8AD 101043841 IC50 = 1300 nM T72458 C1KS2F 101043843 IC50 = 190 nM T72458 CI8PR4 118718122 EC50 = 3.6 nM T72458 CCL46X 118718855 IC50 > 10000 nM T72458 CK6FL5 118718881 EC50 = 14.6 nM T72458 CR13SP 118720353 EC50 = 3.981 nM T72458 CU2D0B 118720354 EC50 = 8.1 nM T72458 C1RU9V 118720355 EC50 = 13 nM T72458 C0WC7Q 118720356 EC50 = 3.7 nM T72458 CCO29V 118720357 EC50 = 24 nM T72458 CQ25BM 118720358 EC50 = 400 nM T72458 CJ3XW9 118720360 EC50 = 1.549 nM T72458 CM24SH 118720361 EC50 = 1.95 nM T72458 CU8DM7 118720362 EC50 = 2.138 nM T72458 C2SNQ7 118720363 EC50 = 1.8 nM T72458 C01ZPV 118720364 EC50 = 1.862 nM T72458 CF2P9J 118720365 EC50 = 4.074 nM T72458 CACO39 118720366 EC50 = 1.95 nM T72458 CI7J4T 118720367 EC50 = 1.585 nM T72458 CSX01G 118720368 EC50 = 1.3 nM T72458 CTJ18H 118720369 EC50 = 1.4 nM T72458 C76NQJ 118720370 EC50 = 1.698 nM T72458 CQ80IN 118720371 EC50 = 82 nM T72458 C4D9HL 118720372 EC50 = 236 nM T72458 CKP1Q6 118720373 EC50 = 188 nM T72458 C71OYW 118720374 EC50 = 11 nM T72458 C8ME0B 118735099 EC50 = 0.3 nM T72458 CK17XF 118735100 IC50 = 6.5 nM T72458 C1O7GU 118735101 EC50 = 0.3 nM T72458 CBTC79 118735102 EC50 = 227 nM T72458 C1O3GL 118735103 IC50 = 200 nM T72458 CAP67E 122178151 IC50 = 70 nM T72458 C65WMB 122184498 IC50 = 2.4 nM T72458 CH9L8O 122184499 IC50 = 18.2 nM T72458 CAQ17N 122184571 IC50 = 16.2 nM T72458 CK48WX 122184572 IC50 = 6.35 nM T72458 CF9PO7 122184573 IC50 = 1390 nM T72458 C3FBZ9 122184574 IC50 = 65.9 nM T72458 CCP0X7 122184575 IC50 = 111 nM T72458 C7OBX1 122184576 IC50 = 1010 nM T72458 CU73AF 122184577 EC50 = 2400 nM T72458 CGB7F4 122184578 IC50 = 134 nM T72458 CB7HZ8 122184579 IC50 = 59.4 nM T72458 C9HE4L 122184580 IC50 = 32.2 nM T72458 C9MJT7 122184581 IC50 = 244 nM T72458 C20NAY 122184582 EC50 = 35.5 nM T72458 CH1B8W 122184631 IC50 = 98 nM T72458 CLXB63 122184632 IC50 = 1700 nM T72458 CIJ14O 122184633 EC50 = 5 nM T72458 CDSR31 122184634 EC50 = 197 nM T72458 CL28BX 122184635 IC50 = 100 nM T72458 CYOR02 122184636 EC50 = 138 nM T72458 C09LFS 122184637 EC50 = 1570 nM T72458 C5CDX9 122184638 EC50 = 946 nM T72458 C64BPZ 122184639 IC50 = 99.9 nM T72458 CEDT39 122184640 EC50 = 1000 nM T72458 CLB43S 122184641 EC50 = 6590 nM T72458 CN4L5U 122184908 EC50 = 0.8 nM T72458 CG0U7B 122184909 EC50 = 152 nM T72458 CZ4HW7 122184910 IC50 = 0.5 nM T72458 C6KW7J 122184911 EC50 = 840 nM T72458 CK3VM5 122184912 EC50 = 1110 nM T72458 C0AFH9 122184913 EC50 = 485 nM T72458 CNBA05 122184914 EC50 = 1450 nM T72458 CARC80 122194229 Ki = 0.14 nM T72458 C80KPB 127046235 EC50 = 0.67 nM T72458 CE63JM 127046977 EC50 = 1.1 nM T72458 CI7TE9 127047209 EC50 = 5.5 nM T72458 C5GX7N 127047475 EC50 = 0.57 nM T72458 C28UAD 127047853 EC50 = 1.2 nM T72458 C9CYP2 127047913 EC50 = 2 nM T72458 C1SF3V 127048118 EC50 = 0.95 nM T72458 CGKE81 132938008 IC50 = 7.5 nM T72458 C7CLU6 133053557 EC50 = 280 nM T72458 CKV0P6 136024005 Ki = 7 nM T72458 CJNF06 137631599 EC50 = 19.95 nM T72458 COM8N7 137631628 IC50 > 1000 nM T72458 CW9P1D 137633115 EC50 = 128 nM T72458 CF2NA9 137633806 EC50 = 1.4 nM T72458 CTD90C 137634090 EC50 = 3800 nM T72458 CPL59T 137635422 EC50 = 1.8 nM T72458 CM1H6A 137636428 EC50 = 677.5 nM T72458 CU4KL7 137636677 EC50 = 602.56 nM T72458 CVC3Q2 137636965 EC50 = 524.81 nM T72458 CK2CZ3 137637026 EC50 = 3.2 nM T72458 CME01A 137637283 EC50 = 0.34 nM T72458 C6TKX9 137637656 EC50 = 2.8 nM T72458 C2FEA6 137638725 EC50 = 6.166 nM T72458 CH17TL 137638778 EC50 = 1.4 nM T72458 CKR14I 137639770 EC50 = 2.1 nM T72458 CHB9X0 137640703 EC50 = 501.19 nM T72458 CBL5Z9 137641157 EC50 = 87.1 nM T72458 CCPD94 137641398 EC50 = 120.23 nM T72458 CTN96O 137642298 EC50 = 71 nM T72458 CGP0V3 137643023 EC50 = 184.6 nM T72458 CAT50J 137643076 EC50 = 178 nM T72458 C5R2TI 137643266 IC50 = 20 nM T72458 CE0YF4 137643385 EC50 = 317.9 nM T72458 C68AYB 137644225 EC50 = 12.7 nM T72458 CJ1I7B 137645567 EC50 > 100000 nM T72458 CKES17 137646333 EC50 = 46773.51 nM T72458 CT18GM 137646617 EC50 = 1047.13 nM T72458 CV5RX4 137647009 EC50 = 6.4 nM T72458 CY7K4J 137647538 EC50 = 114.82 nM T72458 C10VFY 137648144 EC50 = 7.6 nM T72458 C5X7AK 137648344 EC50 = 200 nM T72458 CSF97J 137649543 EC50 = 257.7 nM T72458 CIV6Z7 137649910 EC50 > 3000 nM T72458 CF3VP0 137651074 IC50 = 5 nM T72458 CH62TM 137653176 EC50 > 3000 nM T72458 CF5Z2W 137653739 EC50 = 0.2 nM T72458 CKX3Q9 137653925 EC50 = 1737.8 nM T72458 C12DIK 137655051 Ki = 0.79 nM T72458 CMO01K 137655905 EC50 = 3090.3 nM T72458 CKL0Y8 137656033 EC50 = 112.3 nM T72458 C5WHL4 137656521 EC50 = 11.4 nM T72458 C5FI6X 137657633 IC50 = 45 nM T72458 COS0A1 137658158 EC50 = 147.91 nM T72458 CS1PR7 137659394 EC50 = 478.63 nM T72458 CHB32J 137659790 EC50 = 467.74 nM T72458 CQ7S0L 137659949 EC50 = 21000 nM T72458 C2XLI7 137660671 EC50 = 229.09 nM T72458 C98FVD 137660993 EC50 = 27.54 nM T72458 C4CFP9 137661893 EC50 > 3000 nM T72458 CCZ72V 137662147 EC50 = 2.3 nM T72458 C2WC5J 145948876 IC50 = 950 nM T72458 CUC3S2 145948912 EC50 = 220 nM T72458 C8D7OM 145964017 EC50 = 3.2 nM T72458 CAT7W0 145964349 Ki = 29 nM T72458 CCK75J 145964837 EC50 = 6.7 nM T72458 CS73TM 145966364 EC50 = 1000 nM T72458 CHU51B 145966490 EC50 = 5.3 nM T72458 CJO1Y6 145966716 EC50 = 270 nM T72458 C9RA7Q 145967155 IC50 = 71 nM T72458 CICD84 145971389 EC50 = 150 nM T72458 C97DEG 145971673 EC50 = 720 nM T72458 CEV4F6 145972289 IC50 = 100 nM T72458 C9NRU8 145973779 IC50 = 59 nM T72458 CYD0J5 145973975 IC50 = 73 nM T72458 CR2NQ5 145975465 EC50 = 6.7 nM T72458 CKP26E 145976444 EC50 = 18 nM T72458 C7UJ8Q 145976863 EC50 = 120 nM T72458 CMS17N 145977650 EC50 = 10 nM T72458 CJ28PL 145980198 EC50 = 133 nM T72458 C0S1IN 145980719 EC50 = 928 nM T72458 CEZU78 145980838 IC50 = 2.1 nM T72458 CF34MX 145988152 EC50 = 36 nM T72458 C39KYZ 145988867 EC50 = 280 nM T72458 C7WF3R 145989222 EC50 = 17 nM T72458 C50ZLS 145990599 EC50 = 407 nM T72458 CDQZ25 145994283 IC50 = 10 nM T72458 CE3CN7 155527254 EC50 = 0.03 nM T72458 CX9B4Y 155531854 EC50 = 1.9 nM T72458 C3Q8AU 155532197 EC50 = 5.9 nM T72458 CA5R2L 155532232 IC50 = 14300 nM T72458 C0P7XR 155536962 IC50 = 19300 nM T72458 C6K3AW 155544852 IC50 = 32.2 nM T72458 CQZ7X1 155546131 IC50 = 2700 nM T72458 C7IS0X 155548853 IC50 = 250 nM T72458 CD3J2E 155551202 IC50 = 15700 nM T72458 C20BJD 155551699 EC50 = 4.7 nM T72458 C7C3QR 155551846 EC50 = 0.06 nM T72458 C2SFV9 155561116 IC50 = 1016 nM T72458 CCUT09 155563057 EC50 = 1.9 nM T72458 C1AE7Z 155566718 IC50 = 22000 nM T72458 CR08PO 24858629 IC50 > 1000 nM T72458 D00HAJ 73347136 IC50 = 13000 nM T72458 D00TSX 11672424 IC50 = 100 nM T72458 D00VYC 44400370 EC50 = 0.27 nM T72458 D00XMP 14364677 Ki = 700 nM T72458 D01HTX 11707715 IC50 = 600 nM T72458 D01VMU 44445082 EC50 > 2000 nM T72458 D02JVA 44408515 IC50 = 77 nM T72458 D02MPZ 11535237 EC50 = 2000 nM T72458 D03AZC 25078192 EC50 = 0.16 nM T72458 D04BOG 11629290 IC50 = 150 nM T72458 D04YZZ 44445083 IC50 = 330 nM T72458 D05LLI 11498895 EC50 = 130 nM T72458 D05WNC 11520823 IC50 = 34 nM T72458 D05XRI 44400401 EC50 = 0.26 nM T72458 D05ZUX 44207909 Ki >= 1000 nM T72458 D06PNU 44409257 EC50 = 10 nM T72458 D06RTP 11700730 EC50 = 16 nM T72458 D07DWH 44400402 EC50 = 0.28 nM T72458 D07IBF 44400322 EC50 = 0.54 nM T72458 D07RRN 44406884 Ki = 0.71 nM T72458 D07SFD 44408443 EC50 = 174 nM T72458 D07SRW 10258635 IC50 = 1100 nM T72458 D07UXW 44408400 IC50 = 170 nM T72458 D08DND 44445084 IC50 = 930 nM T72458 D08EBV 44406905 EC50 = 3.2 nM T72458 D09HHW 9842665 IC50 = 103 nM T72458 D09LHF 44413535 EC50 = 16.4 nM T72458 D09OMI 44400400 EC50 = 0.1 nM T72458 D09PDT 24774519 IC50 = 430 nM T72458 D09UUC 46877881 Ki = 190 nM T72458 D09XCH 44400371 EC50 = 5.24 nM T72458 D0A8ME 44400398 EC50 = 0.3 nM T72458 D0B8GR 44413876 EC50 = 5.7 nM T72458 D0B9NH 44408399 EC50 > 10000 nM T72458 D0C7VI 44400369 EC50 = 0.24 nM T72458 D0D8YP 763557 Ki = 2000 nM T72458 D0F6GX 44409240 EC50 = 44 nM T72458 D0GN9K 24774602 IC50 > 10000 nM T72458 D0L1MJ 11700739 IC50 = 16 nM T72458 D0M2QK 44413536 EC50 = 15.4 nM T72458 D0M4EF 11593084 EC50 = 3000 nM T72458 D0N6AS 44158031 EC50 = 200 nM T72458 D0N6KO 9938402 Ki = 0.05 nM T72458 D0P4GI 11629326 IC50 = 1000 nM T72458 D0QW4A 24774356 IC50 = 777 nM T72458 D0R0BY 44400320 EC50 = 0.06 nM T72458 D0R5KO 44413537 Ki = 670 nM T72458 D0T2RY 9948320 Ki >= 1000 nM T72458 D0U1UZ 44413577 EC50 = 1578 nM T72458 D0U5KM 11093672 EC50 = 0.93 nM T72458 D0U6XP 16724004 EC50 = 5700 nM T72458 D0V1JT 9875763 EC50 = 1.25 nM T72458 D0V5YV 44413592 Ki = 4420 nM T72458 D0VD7R 44408408 IC50 = 2700 nM T72458 D0W1SM 44408413 EC50 > 10000 nM T72458 D0WG8P 44400321 EC50 = 0.12 nM T72458 D0WI8M 44445085 IC50 = 300 nM T72458 D0X1YL 25078242 EC50 = 0.92 nM T72458 D0XQ5U 24774438 IC50 > 1000 nM T72458 D0YB7F 92432 EC50 < 0.03162 nM T72458 D0Z1QU 10098971 Ki = 7.9 nM T72458 D0ZD3M 44400399 EC50 = 0.79 nM T16514 D01XNB 4594 Ki = 3400 nM T16514 D03ZFG 5282054 IC50 = 0.19 ug.mL-1 T16514 D04AIT 5280445 IC50 = 62500 nM T16514 D0KL4J 5029 Ki = 5900 nM T16514 D0T6XX 4679 Ki = 4100 nM T16514 D0T9TJ 3034010 Ki = 280 nM T16514 D05TPI 72276 IC50 > 100000 nM T16514 D0U2BH 65064 IC50 = 51970 nM T16514 D0E4WF 439176 Ki = 1500000 nM T16514 C2KJI7 3883 Ki = 5300 nM T16514 CJ0I1N 13792 Ki = 30000 nM T16514 CTHE54 122841 IC50 = 49100 nM T16514 C0WR5N 145691 Ki = 140000000 nM T16514 CCG98V 165114 Ki = 500000 nM T16514 C5Q1JX 182232 IC50 > 1000000 nM T16514 C3FJQ1 485186 IC50 = 91070 nM T16514 CZYL67 2292609 Ki = 380 nM T16514 CMP0Z5 4782471 IC50 = 1140 nM T16514 CE6K3P 5281635 IC50 = 40980 nM T16514 CH01XT 5281656 IC50 = 17850 nM T16514 CJC35O 5282800 IC50 = 100000 nM T16514 CY0CO2 5495925 IC50 = 24830 nM T16514 C51EUJ 7873335 IC50 >= 50000 nM T16514 CG2V5K 7873337 IC50 = 1100 nM T16514 C75GIM 9881506 IC50 = 59000 nM T16514 C9XI1C 9977422 IC50 > 1000 ug.mL-1 T16514 CHZ2D5 9995235 IC50 > 50 ug.mL-1 T16514 C8MXH4 10000563 IC50 > 50 ug.mL-1 T16514 CS7FC2 10020330 IC50 > 50 ug.mL-1 T16514 CTVI84 10040478 IC50 > 50 ug.mL-1 T16514 CNQH21 10040479 IC50 = 2.1 ug.mL-1 T16514 C1PK2F 10044646 IC50 > 1000 ug.mL-1 T16514 CNX5Z8 10085202 IC50 > 50 ug.mL-1 T16514 CUM0N6 10087016 IC50 = 4.6 ug.mL-1 T16514 C9P3CS 10087923 IC50 > 50 ug.mL-1 T16514 C51CUM 10092378 Ki = 30000 nM T16514 C64XGK 10176955 IC50 > 50 ug.mL-1 T16514 CVFJ46 10246217 IC50 > 50 ug.mL-1 T16514 CWI1H5 10266601 IC50 > 50 ug.mL-1 T16514 C5LRW4 10298511 IC50 = 3300 nM T16514 CV6IH8 10354980 IC50 > 50 ug.mL-1 T16514 CVF7Z2 10359032 IC50 = 6.8 ug.mL-1 T16514 C0M2RF 10404949 IC50 > 50 ug.mL-1 T16514 C5MUE3 10422346 IC50 > 50 ug.mL-1 T16514 CQ2LZ5 10466563 IC50 > 50 ug.mL-1 T16514 CJW43Z 10469992 IC50 > 50 ug.mL-1 T16514 C5X7YI 11050315 IC50 > 50 ug.mL-1 T16514 C24UPE 11529878 IC50 > 50 ug.mL-1 T16514 CO96XN 11541428 IC50 = 160 nM T16514 CWQ56J 11543533 Ki = 2500 nM T16514 CZ5N3C 11722353 IC50 > 50 ug.mL-1 T16514 CQY8H4 11724126 IC50 > 50 ug.mL-1 T16514 C7X6DR 11777194 IC50 > 50 ug.mL-1 T16514 CT5D2I 14378645 IC50 = 60200 nM T16514 C45BLU 15081407 IC50 = 31000 nM T16514 C1PJ8I 15788084 Ki = 100000 nM T16514 CO04TC 16046225 IC50 = 25400 nM T16514 CWR7N5 19910294 IC50 = 8590 nM T16514 C19EMT 23649126 IC50 = 160 nM T16514 C9QBC6 25096732 IC50 = 56100 nM T16514 CNCT63 25096734 IC50 = 71700 nM T16514 C06NHT 38390838 IC50 = 50000 nM T16514 CE7B0W 44290695 Ki = 220000 nM T16514 C1QYT0 44388272 IC50 > 50 ug.mL-1 T16514 C0E3PC 44388283 IC50 > 50 ug.mL-1 T16514 CM27AK 44388295 IC50 > 50 ug.mL-1 T16514 C86TYF 44415373 IC50 > 15000 nM T16514 CC3HM1 44415374 IC50 > 15000 nM T16514 C09HMK 44415477 IC50 > 15000 nM T16514 CJA30S 44415496 IC50 > 15000 nM T16514 CF5L3P 44415497 IC50 > 15000 nM T16514 C1VXO4 44415510 IC50 > 15000 nM T16514 CX5KA8 45266261 Ki = 2500000 nM T16514 C3I7XR 51346964 IC50 = 79 nM T16514 CHQW27 52914172 IC50 = 200 nM T16514 CO5AR4 52914173 IC50 = 300 nM T16514 CQCV94 52945061 IC50 = 49160 nM T16514 CIF69A 52948815 IC50 = 14760 nM T16514 CULB62 54706679 IC50 = 19 nM T16514 CYVU49 54712162 IC50 = 136 nM T16514 CQS8R7 54720260 IC50 = 52 nM T16514 CK0IP7 54720261 IC50 = 54 nM T16514 CV4W0R 54720262 IC50 = 194 nM T16514 CS2G5M 54720263 IC50 = 728 nM T16514 CQ9D3F 54720264 IC50 = 68 nM T16514 CR0S7K 54720274 IC50 = 4164 nM T16514 C16TFJ 54720277 IC50 = 734 nM T16514 CJ9A8U 54720280 IC50 = 127 nM T16514 CCG95F 54737895 IC50 = 402 nM T16514 CR0D3L 54737897 IC50 > 15000 nM T16514 C6N2UI 54737898 IC50 > 15000 nM T16514 C7BE1N 54737901 IC50 = 207 nM T16514 CY0F7L 54737905 IC50 = 101 nM T16514 CRWP39 54737909 IC50 > 15000 nM T16514 C6GPH3 54737911 IC50 = 1294 nM T16514 C2KJS4 56658153 IC50 = 1500 nM T16514 CP7IJ5 56658154 IC50 = 580 nM T16514 CK19VO 56661663 IC50 = 420 nM T16514 C0ED9O 56665072 IC50 = 400 nM T16514 CG24JD 56665073 IC50 = 280 nM T16514 C04ZAH 56668685 IC50 = 480 nM T16514 CI51ES 56672028 IC50 = 310 nM T16514 CBYM16 56672029 IC50 = 290 nM T16514 C6NOF0 56675407 IC50 = 1300 nM T16514 C25VNE 56675408 IC50 = 700 nM T16514 CVOA13 56675409 IC50 = 2400 nM T16514 C6W2ZV 56675410 IC50 = 270 nM T16514 CSR3L6 56675411 IC50 = 910 nM T16514 CD5WP7 56678752 IC50 = 1500 nM T16514 CQK16D 56678753 IC50 > 10000 nM T16514 C89BAK 56678754 IC50 = 190 nM T16514 C6XC1K 56678755 IC50 = 530 nM T16514 C2PYZ9 56678756 IC50 > 3000 nM T16514 C53YIK 56678879 IC50 = 420 nM T16514 C54EIB 56682065 IC50 = 2000 nM T16514 C60CNB 56682066 IC50 = 1400 nM T16514 C9U0SZ 56944776 IC50 = 13 nM T16514 C0E2CB 57330203 IC50 = 6 nM T16514 CD3IC4 57519517 IC50 = 15.8 nM T16514 C15LHR 67353959 IC50 = 3 nM T16514 C5IR7A 68288172 IC50 = 430 nM T16514 CQPC84 68288211 IC50 = 40 nM T16514 CXZ9N7 68288384 IC50 = 17 nM T16514 C38ZAK 68288699 IC50 = 85 nM T16514 CK07RI 68288711 IC50 = 70 nM T16514 C9NFH0 68288836 IC50 = 980 nM T16514 C8D6XN 68288941 IC50 = 590 nM T16514 CYF20R 68288944 IC50 = 130 nM T16514 CN38EO 68288981 IC50 = 35 nM T16514 C8NJ1R 68288986 IC50 = 107 nM T16514 C7EP2D 68289020 IC50 = 60 nM T16514 C6BAD8 68289174 IC50 = 60 nM T16514 CO8X9D 68289184 IC50 = 70 nM T16514 C2HJB7 68289227 IC50 = 870 nM T16514 CVRK70 69081490 IC50 = 251 nM T16514 C64OIV 69085357 IC50 = 10 nM T16514 C6O8MS 69166563 IC50 = 50 nM T16514 CCN1K2 70355043 IC50 = 7.9 nM T16514 C3L7MO 70872230 IC50 = 300 nM T16514 C3O8YN 70872278 IC50 = 480 nM T16514 CK56QA 70873969 IC50 = 990 nM T16514 CU0D8S 71460623 IC50 = 10000 nM T16514 CRH37A 71511821 IC50 = 20 nM T16514 CGU2I3 71541605 IC50 > 50000 nM T16514 C5KQG0 71541606 IC50 > 50000 nM T16514 CN6RQ2 71719838 IC50 = 45 nM T16514 CDC29F 72188556 IC50 = 10 nM T16514 C7B2VH 73332466 IC50 = 28 nM T16514 C6ZPL7 73388616 IC50 = 51 nM T16514 CT3N0M 73388705 IC50 = 22 nM T16514 CF40TL 86272214 IC50 = 110 nM T16514 CMDX07 86272688 IC50 = 12 nM T16514 CHU42Z 86272922 IC50 = 3100 nM T16514 CE4A7B 86273159 IC50 = 11 nM T16514 C3WIN2 86273160 IC50 = 10 nM T16514 CWI9H2 86273162 IC50 = 11 nM T16514 CR4O3Z 86273403 IC50 = 110 nM T16514 C0R2KW 86273408 IC50 = 33 nM T16514 C39ZJT 86273883 IC50 = 26 nM T16514 CG40JA 86275336 IC50 > 5000 nM T16514 C4J8CB 86275339 IC50 = 1800 nM T16514 CW0I7F 86275791 IC50 = 350 nM T16514 C1DAT5 86275793 IC50 = 35000 nM T16514 C7U8LK 86275794 IC50 = 50000 nM T16514 CDF60C 89993363 IC50 = 1380 nM T16514 C7H0RS 89993436 IC50 = 32 nM T16514 CP97LB 89993468 IC50 = 41 nM T16514 CCTW25 89993534 IC50 = 550 nM T16514 C9Z3RV 89993608 IC50 = 69 nM T16514 CW2ND1 89993632 IC50 = 33 nM T16514 CUPS02 89993706 IC50 = 23 nM T16514 CRK0M7 89993860 IC50 = 25 nM T16514 C1GH7D 90001554 IC50 = 46 nM T16514 CMUT58 117631954 IC50 = 54 nM T16514 CDV34G 117632261 IC50 = 57 nM T16514 CZK4A6 117632449 IC50 = 69 nM T16514 CPY70A 117992529 IC50 = 360 nM T16514 C8L2AI 117992579 IC50 = 300 nM T16514 CBO57F 117992669 IC50 = 160 nM T16514 CYQ6V8 117992803 IC50 = 460 nM T16514 C29DCG 117992846 IC50 = 1100 nM T16514 CU73WN 117992892 IC50 = 8510 nM T16514 C5EDL1 117992950 IC50 = 33100 nM T16514 CYD3W2 117992981 IC50 = 250 nM T16514 C6GP4I 117992993 IC50 = 590 nM T16514 C7B8NO 117993006 IC50 = 460 nM T16514 COT7W6 117993116 IC50 = 8710 nM T16514 CW82PK 117993126 IC50 = 790 nM T16514 CIK64W 117993152 IC50 = 120 nM T16514 CT09BE 117993175 IC50 = 8910 nM T16514 C1FUZ4 117993412 IC50 = 130 nM T16514 C54FAV 117999149 IC50 = 83 nM T16514 CZT69Y 117999157 IC50 = 30 nM T16514 CC5GD8 117999160 IC50 = 20 nM T16514 CCO89U 117999164 IC50 = 42 nM T16514 C8VLN5 117999171 IC50 = 50 nM T16514 COZ8I6 117999184 IC50 = 200 nM T16514 CN6LZ9 117999235 IC50 = 20 nM T16514 C8PMK6 117999267 IC50 > 10000 nM T16514 C9Y1PD 117999287 IC50 = 300 nM T16514 C5OKI2 118125364 IC50 = 5888.44 nM T16514 CI47HU 118125371 IC50 = 56.23 nM T16514 C9X0KR 118125374 IC50 = 47.86 nM T16514 CZCA13 118125376 IC50 = 490 nM T16514 CP91UC 118125426 IC50 = 160 nM T16514 CYWI47 118125430 IC50 = 41 nM T16514 CC7I0K 118125439 IC50 = 177.83 nM T16514 CH7S8X 118125468 IC50 = 140 nM T16514 CDC75Z 118125490 IC50 = 30.2 nM T16514 C8OPS5 118125499 IC50 = 93.33 nM T16514 C83ZWH 118144180 IC50 = 93 nM T16514 CYI51F 118621498 IC50 = 32 nM T16514 C2OY4N 118621507 IC50 = 97 nM T16514 CFKI50 118621601 IC50 = 90 nM T16514 CUO5I1 118621602 IC50 = 142 nM T16514 CVM6E7 118621647 IC50 = 61 nM T16514 CB5JZ9 118621761 IC50 = 16 nM T16514 CH74OR 118621798 IC50 = 310 nM T16514 C4S1HV 122192508 IC50 = 6 nM T16514 CMNB15 122197394 IC50 = 28700 nM T16514 CY0QH7 122197395 IC50 = 23100 nM T16514 C34DEV 122197396 IC50 = 29700 nM T16514 C9XV2S 122197397 IC50 = 32600 nM T16514 CUT65O 132503175 IC50 = 1500 nM T16514 C1JB6Y 135407178 IC50 > 50 ug.mL-1 T16514 C8T1FY 135410225 IC50 = 4 ug.mL-1 T16514 C75VLC 135432847 IC50 = 5.7 ug.mL-1 T16514 CWK90L 135449011 IC50 > 50 ug.mL-1 T16514 CJD80P 135457983 IC50 > 50 ug.mL-1 T16514 CP8HN9 135488223 IC50 = 8.4 ug.mL-1 T16514 CTH2W0 135503576 IC50 = 2.8 ug.mL-1 T16514 CX8Y7I 135517312 IC50 = 41 ug.mL-1 T16514 CKU80W 135518065 IC50 > 50 ug.mL-1 T16514 CM1HF2 135526950 IC50 > 50 ug.mL-1 T16514 CQK2T3 135535916 IC50 = 8.7 ug.mL-1 T16514 CW0S7A 136102470 IC50 = 49.2 ug.mL-1 T16514 C61AJU 136102471 IC50 > 50 ug.mL-1 T16514 C2NC9L 137633752 IC50 = 3110 nM T16514 CEJO70 137634807 IC50 = 4810 nM T16514 CDT67V 137637200 IC50 = 160 nM T16514 CMSA73 137639962 IC50 = 3980 nM T16514 C1KN9L 137640079 IC50 = 5550 nM T16514 CNVZ89 137640673 IC50 = 3170 nM T16514 C0EY3T 137643629 IC50 = 2610 nM T16514 CWOY74 137647871 IC50 = 8370 nM T16514 CNFP69 137658811 IC50 = 12600 nM T16514 CJQ6B7 137659959 IC50 = 1190 nM T16514 C01KBD 137661456 IC50 = 9560 nM T16514 CZI19P 145960543 IC50 = 590 nM T16514 C19AFT 145961063 IC50 = 170 nM T16514 CW9NJ4 145961301 IC50 = 450 nM T16514 C3AEW6 145962120 IC50 = 36 nM T16514 CG8B1R 145962440 IC50 = 79 nM T16514 CKFR42 145962726 IC50 = 300 nM T16514 C63PUQ 145963234 IC50 = 28 nM T16514 D01WTQ 5495929 IC50 = 40640 nM T16514 D05IWY 5464078 IC50 = 1240 nM T16514 D06PRC 5281650 IC50 = 5540 nM T16514 D09CLP 439155 Ki = 150000 nM T16514 D0B5GC 11349 IC50 > 100000 nM T16514 D0PO8E 6137 Ki > 150000000 nM T16514 D0QP7C 54737894 IC50 = 1403 nM T59604 D02NEH 178024 EC50 = 0.1995 nM T59604 D0BV3J 9804938 IC50 = 22.9 nM T59604 D01HLO 58438464 Ki = 6.607 nM T59604 D05UYQ 15984937 EC50 > 1000 nM T59604 D0LI1C 44469321 IC50 > 30000 nM T59604 D0O1LU 9827407 IC50 = 62.9 nM T59604 D0UO4B 216208 EC50 = 0.9 nM T59604 D0W9VW 11526696 EC50 = 27 nM T59604 D0XH9B 9810101 EC50 = 3 nM T59604 D09TGZ 6918297 IC50 = 15.9 nM T59604 D0A1KU 11683187 Ki = 4400 nM T59604 D0B3CY 121879 Ki = 63 nM T59604 C7Q3IT 328912 IC50 = 1700 nM T59604 CE16YX 753168 IC50 = 8200 nM T59604 C25ZHX 1221269 IC50 = 250 nM T59604 CL5WT1 1744826 IC50 = 180 nM T59604 C1MJA8 2814760 IC50 > 10000 nM T59604 CD2K4M 3153998 Ki = 870 nM T59604 CQ9ZP3 3153999 Ki = 280 nM T59604 C6LAW3 3154000 Ki = 1320 nM T59604 CJ3K0S 3154005 Ki = 2030 nM T59604 CY4I3A 3174463 Ki = 1290 nM T59604 C7QC1D 3180629 Ki = 1370 nM T59604 C0YXV3 3676358 IC50 = 100 nM T59604 CIB78P 5311280 IC50 = 750 nM T59604 CWX3C4 9804743 IC50 = 1.2 nM T59604 C36UOT 9805090 EC50 = 3 nM T59604 CYP42T 9807597 EC50 = 1 nM T59604 C3Q9FN 9827234 EC50 = 10 nM T59604 C91MIV 9848305 EC50 = 986 nM T59604 C75TME 9849592 EC50 = 72 nM T59604 CK0E8G 9868878 EC50 = 7.6 nM T59604 C74HBN 9870965 EC50 = 11.7 nM T59604 C8PFZ1 9875705 EC50 = 1.585 nM T59604 C8BRO3 9876514 Ki = 5 nM T59604 CDB32K 9890375 EC50 = 14 nM T59604 C4BCX8 9890504 EC50 = 1 nM T59604 CPX3E7 9917957 EC50 = 0.34 nM T59604 C8M7BX 9919153 Ki = 6 nM T59604 CMTS32 9950632 EC50 = 30 nM T59604 C4L8RA 9956908 IC50 = 16 nM T59604 C3LV1I 9987037 EC50 = 19.6 nM T59604 CJ7N9H 10005618 EC50 = 3 nM T59604 CSP71U 10006735 EC50 = 6.3 nM T59604 C5X9KF 10026738 EC50 = 16.6 nM T59604 C25PLS 10029990 EC50 = 5 nM T59604 C3JS1K 10032659 EC50 = 7.95 nM T59604 CG2E6X 10100708 EC50 = 69.2 nM T59604 CI0DX4 10118326 EC50 = 1.8 nM T59604 C1Z0XT 10143731 EC50 = 39 nM T59604 C0S8EM 10166594 EC50 = 2.3 nM T59604 CDUZ27 10186158 IC50 = 25.6 nM T59604 C5MRA2 10207327 IC50 = 58 nM T59604 C0O4KL 10209618 EC50 = 7.3 nM T59604 CR5IU4 10210658 EC50 = 16.98 nM T59604 CE3VR7 10253999 Ki = 220 nM T59604 C8RX9I 10280020 EC50 = 0.73 nM T59604 C1E9MX 10323604 EC50 = 1.096 nM T59604 CF27UE 10345516 EC50 = 0.7943 nM T59604 C76XZR 10346217 Ki > 5000 nM T59604 CO16JV 10415000 EC50 = 2.8 nM T59604 CKG7P1 10415364 IC50 = 32 nM T59604 CWM6U8 10506325 EC50 = 6 nM T59604 CP12CV 10530303 IC50 > 10000 nM T59604 CFY90H 10553921 EC50 = 0.7943 nM T59604 CS60ON 10600702 EC50 = 7.5 nM T59604 CO9VJ3 10602640 EC50 = 5 nM T59604 CMW0Z9 10625750 EC50 = 1.585 nM T59604 CL1PH2 10626337 EC50 = 1.995 nM T59604 CW34CO 10699268 IC50 = 55 nM T59604 C9I5HK 10738173 IC50 > 10000 nM T59604 CD91XJ 10745533 EC50 = 18 nM T59604 COU2W4 10746435 IC50 > 2000 nM T59604 C9G2BH 10791616 EC50 = 5 nM T59604 C5Q2WC 10839304 IC50 > 10000 nM T59604 CS8A4G 10864048 IC50 = 185 nM T59604 CPC62E 10907396 IC50 = 337 nM T59604 C5JZW0 10918326 IC50 = 20.1 nM T59604 CTD32I 10929048 IC50 = 228 nM T59604 CS9T3E 10984260 IC50 = 807 nM T59604 CX2S0A 10984270 IC50 = 59.8 nM T59604 CZ0MB4 10994861 IC50 = 807 nM T59604 C06SQO 11016748 IC50 = 16.9 nM T59604 C7PCL0 11114279 IC50 = 213 nM T59604 CSF5J2 11124146 IC50 = 16.2 nM T59604 C6RDO8 11134880 IC50 = 391 nM T59604 C9O4AY 11145720 IC50 = 167 nM T59604 C9ZWB1 11154001 IC50 = 56 nM T59604 CL85TY 11154823 IC50 = 2.8 nM T59604 C19HVQ 11163070 IC50 = 2700 nM T59604 C8C7FK 11166495 IC50 = 83 nM T59604 CQD27L 11176805 IC50 = 67 nM T59604 CVX23I 11178309 IC50 = 70 nM T59604 CX52ZC 11179347 IC50 = 6.9 nM T59604 CB5J8R 11190594 IC50 = 2.8 nM T59604 C9B7QL 11211892 IC50 = 72 nM T59604 C1IQU2 11221946 IC50 = 310 nM T59604 CAG74M 11225576 IC50 = 0.3 nM T59604 CE59SF 11248021 IC50 = 34 nM T59604 C9VA4H 11256439 IC50 = 160 nM T59604 C5QEH2 11258291 EC50 = 40 nM T59604 CTH56E 11281346 IC50 = 50 nM T59604 CIG85H 11282247 IC50 = 19 nM T59604 CZ12BJ 11306502 EC50 = 0.46 nM T59604 CI28KO 11314908 IC50 = 221 nM T59604 CXT20O 11327400 IC50 = 86 nM T59604 CVU6P9 11328064 IC50 = 120 nM T59604 C1H5CL 11328920 IC50 = 2 nM T59604 C5M3ZN 11329138 IC50 = 29 nM T59604 C7Y8VZ 11337482 IC50 = 11 nM T59604 C5A7VJ 11339816 IC50 = 1.5 nM T59604 C7QV2P 11340044 IC50 = 5.8 nM T59604 CI2TD8 11340329 IC50 = 7 nM T59604 C85DMO 11349789 IC50 = 66 nM T59604 C3FID2 11351838 IC50 = 10 nM T59604 C79PWN 11353414 EC50 = 1.5 nM T59604 C23YMZ 11373823 IC50 = 126 nM T59604 CX21SG 11410373 IC50 = 0.4 nM T59604 C5ZH0O 11430392 IC50 = 4.2 nM T59604 C4EL7T 11430583 IC50 = 37 nM T59604 C38KZA 11431274 IC50 = 0.4 nM T59604 C02SXV 11441978 IC50 = 11 nM T59604 CH8IF2 11442040 IC50 = 88 nM T59604 C41XHB 11452801 IC50 = 18 nM T59604 CV0M3Q 11453509 IC50 = 7.7 nM T59604 C6IJ8W 11454617 IC50 = 2.5 nM T59604 CJS58R 11455251 IC50 = 137 nM T59604 CF81ZH 11476589 IC50 = 0.8 nM T59604 C09NWX 11503585 IC50 = 308 nM T59604 CA6BI9 11508639 IC50 = 300 nM T59604 CB7VA3 11517629 IC50 = 37 nM T59604 CSB20C 11523411 IC50 = 110 nM T59604 CDOF50 11525404 EC50 = 10 nM T59604 CG3AZ5 11531313 IC50 = 550 nM T59604 CYO8E0 11532288 EC50 = 15.85 nM T59604 CGS1J2 11537683 IC50 = 110 nM T59604 C5F8WZ 11537800 IC50 = 57 nM T59604 C3ROC9 11538533 IC50 = 7 nM T59604 C6Z4IU 11538534 IC50 = 9.8 nM T59604 CU4AY2 11539587 IC50 = 492 nM T59604 CD2TQ8 11539588 IC50 = 861 nM T59604 CLG67J 11539642 EC50 = 2.512 nM T59604 C17VJD 11554351 EC50 = 39.81 nM T59604 CGY7Z8 11556936 IC50 = 8530 nM T59604 C87NYP 11556937 IC50 = 15700 nM T59604 CPK5I8 11568561 IC50 = 600 nM T59604 CTWI32 11576186 EC50 = 15.85 nM T59604 CI3LV0 11576960 IC50 = 98 nM T59604 CJ1RE7 11577349 IC50 = 10 nM T59604 CZY1F4 11582836 IC50 = 410 nM T59604 CR87OJ 11583811 IC50 = 2.9 nM T59604 CP07SD 11584048 EC50 = 0.7943 nM T59604 C2PS0V 11605061 EC50 = 39.81 nM T59604 C8LS5D 11605333 IC50 = 5.7 nM T59604 C83JXN 11605822 IC50 = 25 nM T59604 C3Q0JA 11606121 IC50 = 4900 nM T59604 CL9E5D 11612155 IC50 = 6.3 nM T59604 CAX29H 11617435 IC50 = 290 nM T59604 CO0X6G 11618705 IC50 = 53 nM T59604 C0PE7U 11626181 IC50 = 319 nM T59604 C2Z5OD 11633712 EC50 = 100 nM T59604 C3UW1I 11646276 IC50 = 9.2 nM T59604 CEA68R 11649239 IC50 = 18 nM T59604 C8JQ6X 11649248 IC50 = 39 nM T59604 C7A6DM 11654867 IC50 = 3350 nM T59604 C5X9KU 11655355 IC50 = 320 nM T59604 C6YW9T 11655578 IC50 = 780 nM T59604 CCYT36 11662746 EC50 = 63.1 nM T59604 CF0WK6 11663710 IC50 = 8 nM T59604 CL14RB 11669486 IC50 = 41 nM T59604 CF14EQ 11676995 IC50 = 110 nM T59604 C4MRC3 11677781 IC50 = 19 nM T59604 C42VAZ 11683469 IC50 = 2.4 nM T59604 C8VTS6 11690097 IC50 = 3.7 nM T59604 C61WEI 11692087 IC50 = 6 nM T59604 CE0F1A 11697618 IC50 = 280 nM T59604 C3X4IJ 11699004 IC50 = 57 nM T59604 CM9WV4 11712108 EC50 = 6.31 nM T59604 CW34HT 11712151 IC50 = 1.2 nM T59604 CQL7H2 11713497 IC50 = 9 nM T59604 CGZ57K 11731384 IC50 = 116 nM T59604 CVS7D5 11751384 IC50 = 343 nM T59604 CBK20C 11827047 IC50 = 22.7 nM T59604 C9XI4T 11846463 IC50 = 11 nM T59604 CWP0B9 11846624 IC50 = 109 nM T59604 CCUF60 11846625 IC50 = 249 nM T59604 CF6D4C 11846627 IC50 = 2270 nM T59604 C5D4KB 11846628 IC50 = 1670 nM T59604 CJ3AT5 11846629 IC50 = 391 nM T59604 CD4VX3 11846630 IC50 = 3080 nM T59604 CWSA56 11846799 IC50 > 1000 nM T59604 CQ9FO0 11846800 IC50 > 10000 nM T59604 C6C8DJ 15481181 EC50 = 3 nM T59604 CJ3SG7 15481185 EC50 = 3.981 nM T59604 C9STQ7 15481188 EC50 = 3 nM T59604 COA2U1 15945877 IC50 = 11 nM T59604 COZU71 15949382 IC50 = 54 nM T59604 C20CRP 16040587 EC50 = 100 nM T59604 C8ZP3G 16041292 EC50 = 501.19 nM T59604 CR0JL5 16112909 IC50 = 660 nM T59604 CJB54V 16112910 IC50 = 560 nM T59604 CD85OU 16112911 IC50 = 750 nM T59604 CA5D3X 16113002 IC50 = 38 nM T59604 COF94S 16113003 IC50 = 5.6 nM T59604 CQ59HR 16113122 IC50 = 154 nM T59604 C8MU4Z 16113124 IC50 = 828 nM T59604 C6K7IZ 16113245 IC50 = 4.5 nM T59604 C96CEF 16113246 IC50 = 8 nM T59604 C2ZGY6 16113248 EC50 = 7.7 nM T59604 C6TGZ4 16113370 IC50 = 29 nM T59604 CDC6B4 16113371 EC50 = 6 nM T59604 CRV2T0 16113372 IC50 = 28 nM T59604 CMSC45 16113468 IC50 = 108 nM T59604 CUJ3A6 16113469 IC50 = 80 nM T59604 CBW76F 16113471 IC50 = 100 nM T59604 CB0J6E 16113472 IC50 = 200 nM T59604 CBU67D 16113474 IC50 = 850 nM T59604 C9IQZ5 16113577 EC50 = 15 nM T59604 CG3H1E 16113578 IC50 = 220 nM T59604 CQ8Z4O 16113579 IC50 = 125 nM T59604 CTI61R 16113580 EC50 = 4 nM T59604 C3OGV4 16113581 IC50 = 120 nM T59604 C7H2GA 16113582 IC50 = 1700 nM T59604 CL98BH 16113583 IC50 = 580 nM T59604 CIQ6S3 16113584 IC50 = 2200 nM T59604 CD85FI 16113585 IC50 = 1000 nM T59604 C95IGA 16113691 IC50 = 15 nM T59604 C0A6WM 16113692 EC50 = 49 nM T59604 C4YLV6 16113693 EC50 = 18 nM T59604 CJ0D5P 16113694 IC50 = 140 nM T59604 C2T4OR 16113695 IC50 = 6 nM T59604 CJ43OU 16113710 EC50 = 5.4 nM T59604 C85YDF 16113796 IC50 = 120 nM T59604 CFQP15 16113797 IC50 = 150 nM T59604 C7U9GO 16113798 IC50 = 150 nM T59604 C6JU3V 16113799 IC50 = 83 nM T59604 CR63OJ 16113800 EC50 = 45 nM T59604 CQ02OX 16113902 IC50 = 11 nM T59604 CVO4T3 16113903 IC50 = 150 nM T59604 C9KMB0 16113904 IC50 = 12 nM T59604 CY29UJ 16113905 IC50 = 145 nM T59604 CFR8D6 16113906 EC50 = 140 nM T59604 C6OXS9 16114008 IC50 = 56 nM T59604 CFY8I0 16114009 IC50 = 130 nM T59604 CF16SW 16114010 IC50 = 55 nM T59604 CY2W6P 16114011 EC50 = 210 nM T59604 CJ4I2K 16114012 IC50 = 170 nM T59604 CM1LX9 16114096 IC50 = 0.5 nM T59604 C5U8PQ 16114097 EC50 = 5.3 nM T59604 CD9C6M 16114098 EC50 = 12 nM T59604 CO1QH0 16114099 IC50 = 28 nM T59604 C7IHG1 16114181 IC50 = 140 nM T59604 C58OIJ 16114183 IC50 > 1000 nM T59604 C4GV2E 16114184 IC50 = 173 nM T59604 CEH6N4 16114289 IC50 = 7 nM T59604 CRT04N 16114290 EC50 = 11 nM T59604 C1DS8N 16114292 IC50 = 0.3 nM T59604 CHQ5N8 16114403 IC50 = 23 nM T59604 CI0PQ3 16114404 IC50 = 32 nM T59604 CE4ZJ1 16114514 EC50 = 9.9 nM T59604 C3N6GQ 16114530 IC50 = 195 nM T59604 CFR8P6 16114531 IC50 = 240 nM T59604 CF0AE8 16114532 IC50 = 96 nM T59604 CSF23I 16134923 IC50 = 0.25 nM T59604 CSK20B 16202767 IC50 = 840 nM T59604 CHV75A 16203236 IC50 = 570 nM T59604 C5D0OB 16203237 EC50 = 23 nM T59604 CRTW49 16203238 EC50 = 41 nM T59604 C6KMR5 16203349 IC50 = 550 nM T59604 C9BHK2 16203569 IC50 = 62 nM T59604 C7U5FV 16203571 IC50 > 1000 nM T59604 CSH9C8 16203918 IC50 = 440 nM T59604 C8QC3F 16203930 IC50 = 110 nM T59604 C6UBC9 16204021 IC50 = 400 nM T59604 CPHM06 16204037 IC50 = 410 nM T59604 CE7Q6B 16204131 IC50 > 1000 nM T59604 CTQD10 16204133 IC50 > 1000 nM T59604 CIQU08 16204145 IC50 = 500 nM T59604 C4R7IG 16204226 IC50 = 470 nM T59604 CS28IM 16204229 IC50 = 700 nM T59604 CS70IJ 16204237 IC50 = 640 nM T59604 CZX82H 16204239 IC50 = 300 nM T59604 CD9A5X 16204241 IC50 = 310 nM T59604 C4SJB9 16204336 IC50 > 1000 nM T59604 CQD54B 16204343 IC50 = 640 nM T59604 CB7RM8 16204433 IC50 > 1000 nM T59604 C1D9TP 16752684 EC50 = 0.1585 nM T59604 C4AZ3J 16752689 EC50 = 125.89 nM T59604 CV46HZ 20600693 EC50 = 0.85 nM T59604 CXS09R 22862436 EC50 = 5 nM T59604 CWR42Q 22867441 EC50 = 0.6 nM T59604 CX8W0F 22888352 EC50 = 2 nM T59604 CXLY27 22888359 EC50 = 9.8 nM T59604 C4QSI5 22888379 EC50 = 19.7 nM T59604 CR01IA 22888395 EC50 = 7.6 nM T59604 CD5Y1W 22888424 EC50 = 3.4 nM T59604 C9XC7B 22888425 EC50 = 5.6 nM T59604 COJ8D5 22888428 EC50 = 14.4 nM T59604 CLYK60 22888433 EC50 = 4.9 nM T59604 CM1D8Q 22888474 EC50 = 0.46 nM T59604 C5X3IN 22888475 EC50 = 1.4 nM T59604 CZ3JV2 22888476 EC50 = 0.49 nM T59604 CL2XZ6 22888486 EC50 = 12 nM T59604 C7H6MC 23631026 EC50 = 6.5 nM T59604 CQ1M3P 23631387 IC50 = 52 nM T59604 CHU29W 23635235 Ki = 680 nM T59604 C5NO7V 23648232 IC50 = 759 nM T59604 CO2KQ7 23648233 IC50 > 1000 nM T59604 CCV54W 23648234 IC50 > 1000 nM T59604 CL3KB7 23648235 IC50 > 1000 nM T59604 CCER83 23648236 EC50 = 279 nM T59604 C0PJ1C 23648242 IC50 = 350 nM T59604 C0OPG8 23648244 EC50 = 2.5 nM T59604 C2EBF7 23648245 IC50 = 16 nM T59604 CNFQ62 23648246 IC50 = 130 nM T59604 C6EGQ3 23648249 EC50 = 2.3 nM T59604 CD0G8V 23648250 EC50 = 15 nM T59604 CAUC58 23649669 EC50 = 1.9 nM T59604 C73PIU 23656300 IC50 = 134 nM T59604 C8KO9M 23661656 EC50 = 4100 nM T59604 CU4T8D 23730225 EC50 = 3 nM T59604 CE3UN2 23730226 EC50 = 5.5 nM T59604 CD5U2Z 23730227 EC50 = 14.6 nM T59604 C1KX8D 23730228 EC50 = 3.8 nM T59604 C1YFU5 23730339 EC50 = 10.1 nM T59604 CK40WD 23730340 EC50 = 82.5 nM T59604 C4M6IA 23730341 EC50 = 3.3 nM T59604 CU7PS4 23730342 EC50 = 7.9 nM T59604 C69RSP 23730343 EC50 = 9.5 nM T59604 CG6TP5 23730458 EC50 = 45.3 nM T59604 CK2Q5J 24180592 Ki = 460 nM T59604 C7SMW5 24180646 EC50 = 79 nM T59604 C60NCW 24755624 EC50 = 0.7943 nM T59604 CU9B7S 24803347 EC50 = 3.981 nM T59604 C09HSR 24894012 EC50 = 0.27 nM T59604 C0P5DO 25010378 EC50 = 0.2 nM T59604 CHX91V 25022503 EC50 = 1.18 nM T59604 CCTG60 25022506 EC50 = 3.981 nM T59604 CMU30E 25022640 EC50 = 0.4 nM T59604 CK0X9U 25032438 Ki = 15 nM T59604 CY6DL8 25098836 EC50 = 2 nM T59604 CV9KH6 25190330 IC50 > 10000 nM T59604 CN35SM 25190383 Ki = 44 nM T59604 CH8RI6 25195191 EC50 > 5011.87 nM T59604 C62QAO 25195192 EC50 > 5011.87 nM T59604 CML1Y2 25211977 EC50 = 4 nM T59604 C3SYE2 25227441 IC50 = 0.078 nM T59604 C83ATJ 25260745 IC50 = 0.43 nM T59604 CZ49UK 25260749 IC50 = 0.31 nM T59604 C89RDC 25260900 IC50 = 2.9 nM T59604 CNR21Q 25260901 IC50 = 6.7 nM T59604 C3JB4O 25261382 IC50 = 1.3 nM T59604 C0BZJ4 25262608 IC50 = 44 nM T59604 CU64LE 25262771 IC50 = 27 nM T59604 C9AQI6 25262772 IC50 = 83 nM T59604 CAT4S5 42624368 IC50 > 2000 nM T59604 CW07AM 44235473 IC50 = 2770 nM T59604 CA1S7F 44281449 EC50 = 2.291 nM T59604 C6TEG2 44281450 EC50 = 4.467 nM T59604 C4DL8B 44281466 EC50 = 14.13 nM T59604 CM2PN4 44293091 EC50 = 21.88 nM T59604 CNT64H 44293557 EC50 = 10 nM T59604 CNDR48 44301387 EC50 = 378.1 nM T59604 C8BYR7 44301389 EC50 = 68.2 nM T59604 CC6XA2 44301462 EC50 = 448.5 nM T59604 C8RVG9 44301510 EC50 = 72 nM T59604 CPY84C 44301512 EC50 = 432.2 nM T59604 C35FWU 44336274 IC50 = 0.2 nM T59604 C7RNU6 44340007 Ki = 18 nM T59604 CY3KR2 44340008 Ki = 0.34 nM T59604 CS2V6M 44340268 Ki = 0.45 nM T59604 CNP5Q7 44357681 IC50 = 7.1 nM T59604 C53YHV 44368295 IC50 = 13.2 nM T59604 CE1V6K 44378837 IC50 = 67 nM T59604 CATD24 44378979 IC50 = 960 nM T59604 C9PZX8 44378981 IC50 = 200 nM T59604 C3MI5R 44378986 IC50 = 340 nM T59604 CK02CW 44379034 IC50 = 340 nM T59604 CF75ZD 44379072 IC50 = 1400 nM T59604 C2TR3U 44379301 IC50 = 3500 nM T59604 CKX5P3 44379303 IC50 = 48 nM T59604 CR40BF 44383343 IC50 = 190 nM T59604 CH20JT 44389131 IC50 = 4100 nM T59604 C0A3JZ 44389151 IC50 = 1900 nM T59604 CRP5G3 44389167 IC50 = 6300 nM T59604 CJD5A3 44389168 IC50 = 2200 nM T59604 CUND20 44389186 IC50 = 4000 nM T59604 CC59YF 44389187 IC50 = 18500 nM T59604 CC7B0N 44389192 IC50 = 860 nM T59604 CDX43V 44389215 IC50 = 6000 nM T59604 C7IT1W 44389216 IC50 = 4500 nM T59604 CG4IP9 44389221 IC50 > 10000 nM T59604 C8S2FN 44389222 IC50 > 10000 nM T59604 CS32WV 44389243 IC50 = 7500 nM T59604 C14EAB 44389248 IC50 = 3100 nM T59604 C6H5JB 44389249 IC50 > 10000 nM T59604 CV2LI4 44389262 IC50 = 1200 nM T59604 CAYW89 44389268 IC50 > 10000 nM T59604 CNU50S 44389271 IC50 > 100 nM T59604 C9HM6U 44389278 IC50 > 10000 nM T59604 CB7XS3 44389283 IC50 = 4700 nM T59604 CU57FZ 44390840 IC50 = 1.6 nM T59604 CRWC94 44390849 IC50 = 0.02 nM T59604 CMSQ24 44390860 IC50 = 15 nM T59604 C8P3CZ 44390862 IC50 = 0.24 nM T59604 C0LN3A 44390869 IC50 = 83 nM T59604 CXI52Q 44390871 IC50 = 4.2 nM T59604 C1E5LM 44390881 IC50 = 160 nM T59604 CJ7EY2 44390888 IC50 = 116 nM T59604 C56AGM 44390889 IC50 = 77 nM T59604 CYD1Q9 44390901 IC50 = 106 nM T59604 CEGR27 44390905 EC50 = 21 nM T59604 C85VNO 44390906 EC50 = 257 nM T59604 CMSB67 44390914 EC50 = 3.4 nM T59604 C76FQD 44390922 EC50 = 6.4 nM T59604 CPLC95 44390980 EC50 < 5 nM T59604 CD5O4B 44390986 EC50 = 2.1 nM T59604 CYLP68 44390996 EC50 = 1.5 nM T59604 CPMY25 44390997 EC50 = 41 nM T59604 CZYL89 44391002 EC50 = 20.9 nM T59604 CTNM61 44391003 EC50 = 17.8 nM T59604 CFXO86 44391007 EC50 = 190 nM T59604 CUX58C 44391008 EC50 = 19.6 nM T59604 C9TWS4 44391010 EC50 = 2.4 nM T59604 CJ8G3Y 44391015 EC50 = 45 nM T59604 CE90XM 44391020 EC50 = 27 nM T59604 C4RCW7 44391021 EC50 = 9.2 nM T59604 CBE9S6 44391024 EC50 = 9 nM T59604 CR1KY8 44391027 EC50 = 26.7 nM T59604 C4BZ3X 44391028 EC50 = 257 nM T59604 CVD75K 44391032 EC50 = 4.3 nM T59604 C3MG7O 44391035 EC50 = 43 nM T59604 CCL8I5 44391038 EC50 = 13.1 nM T59604 CDC4G0 44391039 EC50 = 0.66 nM T59604 CQ8GA6 44391040 EC50 = 21 nM T59604 C0R6JA 44391041 EC50 = 7.3 nM T59604 C0G2HS 44391048 EC50 = 219 nM T59604 CUTM09 44394833 IC50 = 15 nM T59604 C13ITZ 44394913 IC50 = 714 nM T59604 C0R3PY 44394930 IC50 = 162 nM T59604 C85FXK 44394947 IC50 = 47 nM T59604 CPI02V 44394974 IC50 = 29 nM T59604 CN76GO 44394982 IC50 = 3 nM T59604 C6R8ZF 44395002 IC50 = 139 nM T59604 CQ3SF5 44395020 IC50 = 103 nM T59604 CHB16Y 44396269 Ki = 1180 nM T59604 C32LQZ 44396306 Ki = 1920 nM T59604 C6VMK1 44396320 Ki = 910 nM T59604 CBJ45U 44396377 Ki = 1170 nM T59604 CNMA04 44396381 Ki = 1150 nM T59604 C6K1UW 44396384 Ki = 2630 nM T59604 C8JL9Z 44409455 IC50 = 690 nM T59604 CFEN21 44409536 IC50 = 1 nM T59604 CVS16R 44409611 IC50 = 137 nM T59604 CEU2B7 44409661 IC50 = 14 nM T59604 CLG34S 44409666 IC50 = 21 nM T59604 C85OXL 44409667 IC50 = 36 nM T59604 C42SDG 44409672 IC50 = 2.7 nM T59604 C0UEZ5 44409673 IC50 = 3.4 nM T59604 CB26CT 44409678 IC50 = 187 nM T59604 CE3P5U 44409679 IC50 = 3430 nM T59604 C6Z4TD 44409683 IC50 = 316 nM T59604 CL5QG4 44409684 IC50 = 5.5 nM T59604 CXP53Z 44409756 IC50 = 1.5 nM T59604 CT3EZ2 44409757 IC50 = 10 nM T59604 CID79S 44409758 IC50 = 5.4 nM T59604 CTH5F1 44409761 IC50 = 2480 nM T59604 CUA64R 44409762 IC50 = 354 nM T59604 C4P7RB 44409763 IC50 = 38 nM T59604 C75DFK 44409764 IC50 = 96 nM T59604 CY7H4Q 44409767 IC50 = 601 nM T59604 C7H9NR 44409770 IC50 = 66 nM T59604 CVP0N3 44409771 IC50 = 283 nM T59604 CLFC80 44409775 IC50 = 32 nM T59604 C20LGI 44409776 IC50 = 10 nM T59604 CBJ25N 44409785 IC50 = 57 nM T59604 CD84BX 44409801 IC50 = 11 nM T59604 CN5M7P 44409802 IC50 = 19 nM T59604 C8EDJ9 44409809 IC50 = 6 nM T59604 CXP6Z1 44409810 IC50 = 82 nM T59604 C5KD8R 44409821 IC50 = 2 nM T59604 CSGL98 44409831 IC50 = 180 nM T59604 CMU4O8 44409832 IC50 = 634 nM T59604 CGFX78 44409839 IC50 = 279 nM T59604 CJHO48 44409840 IC50 = 13 nM T59604 C9RMI5 44409864 IC50 = 69 nM T59604 CB3L8E 44409865 IC50 = 34 nM T59604 CPIF36 44409867 IC50 = 700 nM T59604 C3XY1N 44409868 IC50 = 248 nM T59604 C5BI1G 44409871 IC50 = 186 nM T59604 C28HBI 44409872 IC50 = 3250 nM T59604 C7TGZ8 44409946 IC50 = 41 nM T59604 CPHK59 44409975 IC50 = 69 nM T59604 CMFX65 44409979 IC50 = 192 nM T59604 CRXW67 44409980 IC50 = 244 nM T59604 CYW24G 44409989 IC50 = 38 nM T59604 CIM85O 44409990 IC50 = 5.2 nM T59604 CCHW29 44409994 IC50 = 19 nM T59604 C1Y9BM 44409998 IC50 = 7.5 nM T59604 C5Y6ZL 44410003 IC50 = 61 nM T59604 CE3AK8 44410007 IC50 = 65 nM T59604 CHS4P3 44410008 IC50 = 380 nM T59604 C5O2EZ 44410012 IC50 = 151 nM T59604 CY90GP 44410013 IC50 = 276 nM T59604 CM8NS3 44411584 EC50 = 4.786 nM T59604 CX8UH6 44411632 EC50 = 5.6 nM T59604 C7IF5J 44411634 EC50 = 2.089 nM T59604 CM5W7O 44411718 EC50 = 10 nM T59604 C4XRF0 44411720 EC50 = 8.5 nM T59604 C0EJN5 44411745 EC50 = 2 nM T59604 C4XQN6 44411753 EC50 = 2.692 nM T59604 CD67ZN 44411902 EC50 = 8.5 nM T59604 C8T3EY 44411905 EC50 = 6 nM T59604 CIWC39 44411913 EC50 = 57 nM T59604 CWQC39 44411920 EC50 = 1.3 nM T59604 C74FRH 44421230 IC50 = 520 nM T59604 CZXM91 44433201 IC50 > 1000 nM T59604 C0BAW6 44433202 IC50 > 1000 nM T59604 CO8MG3 44434007 EC50 = 43 nM T59604 CB8TW6 44434008 EC50 = 55 nM T59604 CKE95S 44434009 EC50 = 42 nM T59604 CBX24U 44434010 EC50 = 30 nM T59604 CPDS49 44434011 EC50 = 51 nM T59604 CHJD74 44434012 EC50 = 27 nM T59604 CBL0Q1 44434015 EC50 = 59 nM T59604 CH9T4L 44434016 EC50 = 49 nM T59604 CS5F1U 44434018 EC50 = 200 nM T59604 CV98TX 44434050 EC50 = 99 nM T59604 CTK43V 44434051 EC50 = 1120 nM T59604 CZCP60 44434052 EC50 = 259 nM T59604 CVBI34 44434053 EC50 = 116 nM T59604 CEKD38 44434054 EC50 = 868 nM T59604 CG0SE7 44434055 EC50 = 390 nM T59604 CR6K8O 44434056 EC50 = 426 nM T59604 C4SFH9 44434073 EC50 = 67 nM T59604 CA71NP 44434074 Ki = 2660 nM T59604 CEX1G5 44434076 EC50 = 147 nM T59604 C7XAT2 44434078 EC50 = 546 nM T59604 C4GZ7L 44434080 EC50 = 17 nM T59604 CN89OI 44434083 EC50 = 12 nM T59604 CDX6Z2 44434086 EC50 = 517 nM T59604 C17XZF 44434109 EC50 = 14 nM T59604 CM50KA 44434110 EC50 = 107 nM T59604 CRJB42 44434111 EC50 = 4 nM T59604 C93WND 44434112 EC50 = 150 nM T59604 C1RW8J 44434113 EC50 = 20 nM T59604 CG5BQ6 44434114 EC50 = 3170 nM T59604 CPW7T6 44434118 EC50 = 75 nM T59604 CM9S2J 44434119 EC50 = 347 nM T59604 C1IYT7 44434120 EC50 = 10 nM T59604 CVX30L 44434121 EC50 = 35 nM T59604 C47WIA 44434122 EC50 = 1860 nM T59604 CYP14C 44434123 EC50 = 29 nM T59604 CG5HP6 44434124 EC50 = 1520 nM T59604 C4G7MZ 44436807 IC50 = 138 nM T59604 C0V5AB 44436812 IC50 = 113 nM T59604 C1IZJ3 44436813 IC50 = 275 nM T59604 CHY84U 44436816 EC50 = 256 nM T59604 CBK90A 44436817 IC50 = 175 nM T59604 CE6HN1 44436828 IC50 = 9.5 nM T59604 C91XJV 44436829 IC50 = 32 nM T59604 CLK31M 44436831 IC50 = 44 nM T59604 C7YOX1 44436832 IC50 = 490 nM T59604 CV3KT1 44436833 IC50 > 1000 nM T59604 CB9Y1W 44436842 IC50 = 53 nM T59604 C4ON6U 44436850 EC50 = 1.6 nM T59604 C9FI7B 44436857 EC50 = 6.1 nM T59604 CGW4J7 44436868 IC50 = 468 nM T59604 C5XF8N 44436876 EC50 = 14 nM T59604 C9HWR1 44436881 IC50 = 255 nM T59604 CS49IW 44436882 EC50 = 183 nM T59604 C0B3MG 44436883 EC50 = 8.7 nM T59604 C3YWE7 44436884 EC50 = 12 nM T59604 CF7IT3 44436885 IC50 = 32 nM T59604 CRWI83 44436886 EC50 = 19.6 nM T59604 CAIF68 44436887 EC50 = 143 nM T59604 C1VO4A 44436888 IC50 = 6 nM T59604 CTKA41 44436889 IC50 = 18 nM T59604 C2HRY9 44436917 IC50 = 375 nM T59604 CTE08W 44437953 EC50 = 6.026 nM T59604 CU7W5D 44437955 EC50 = 1 nM T59604 CC8L3E 44437963 EC50 = 77 nM T59604 C4YDC1 44437966 EC50 = 30 nM T59604 CD25BO 44437969 EC50 = 30 nM T59604 C8J1OH 44437971 EC50 = 18 nM T59604 CE2S0F 44437979 EC50 = 0.28 nM T59604 CM8AY5 44444556 EC50 = 158.49 nM T59604 CW9LC3 44444557 EC50 = 125.89 nM T59604 CXYK84 44444558 EC50 = 39.81 nM T59604 C5GHI6 44444559 EC50 = 0.5012 nM T59604 CVL75O 44444560 EC50 = 31.62 nM T59604 CH8N6W 44444562 EC50 = 5.012 nM T59604 C2L6RI 44444563 EC50 = 0.1995 nM T59604 CA0EX4 44444564 EC50 = 19.95 nM T59604 CE4W5D 44444565 EC50 = 2.512 nM T59604 C6RI1A 44444566 EC50 = 3.162 nM T59604 CE5RN2 44444568 EC50 = 3.981 nM T59604 C7L8OG 44444570 EC50 = 63.1 nM T59604 C4YI8W 44444571 EC50 = 0.7943 nM T59604 CY5QN2 44444572 EC50 = 10 nM T59604 C15MKG 44444574 EC50 = 15.85 nM T59604 CE24TG 44445591 IC50 = 108 nM T59604 C4K1JA 44445592 IC50 = 11 nM T59604 CXS78T 44445593 IC50 = 60 nM T59604 C6RLF1 44445594 IC50 = 1.8 nM T59604 C0OB9Q 44445595 IC50 = 1.1 nM T59604 C4O3TW 44445596 IC50 = 33 nM T59604 C6WI0J 44445597 IC50 = 67 nM T59604 CVC8D2 44445598 IC50 = 49 nM T59604 C8BHU7 44445599 IC50 = 1.9 nM T59604 C8CQS1 44445600 IC50 = 0.7 nM T59604 CVDM94 44445601 IC50 = 105 nM T59604 CA7N0D 44445602 IC50 = 160 nM T59604 CS6JW0 44445603 IC50 = 58 nM T59604 CRT76Q 44445604 IC50 > 1000 nM T59604 CF9J8O 44445605 IC50 = 220 nM T59604 CDK82Q 44445606 IC50 = 34 nM T59604 C49ITN 44445607 IC50 = 120 nM T59604 CE8L5D 44445608 IC50 = 51 nM T59604 C96PSH 44445609 IC50 = 96 nM T59604 CWIY32 44445610 IC50 = 7.9 nM T59604 C7OD1G 44445611 IC50 = 3 nM T59604 C6H2AN 44445612 IC50 = 61 nM T59604 CH8O1Q 44445613 IC50 = 700 nM T59604 CSQ18J 44445614 IC50 = 480 nM T59604 CZW47S 44445615 IC50 = 29 nM T59604 CW08EF 44445616 IC50 = 76 nM T59604 C0YMX6 44445617 IC50 = 270 nM T59604 CH35WJ 44445618 IC50 = 177 nM T59604 CL5SN1 44445619 IC50 = 80 nM T59604 C1K4HU 44445620 EC50 = 16 nM T59604 CM09WI 44445621 IC50 > 1000 nM T59604 C3FJX6 44445622 IC50 = 112 nM T59604 C18GVK 44445624 IC50 = 140 nM T59604 C9C2VA 44445625 IC50 = 18.5 nM T59604 CL7VY1 44445626 IC50 = 5 nM T59604 C5W0YR 44445627 IC50 = 14 nM T59604 CPT7N8 44445628 IC50 = 89 nM T59604 C2H8TW 44445629 IC50 = 300 nM T59604 CP1QF3 44446137 IC50 = 140 nM T59604 C2WYK3 44446140 IC50 > 1000 nM T59604 CE3G4V 44446143 IC50 > 1000 nM T59604 C7WZ6E 44446148 IC50 = 450 nM T59604 C3UM2W 44446150 IC50 > 1000 nM T59604 CP73DI 44446152 IC50 > 1000 nM T59604 CCON73 44446154 IC50 > 1000 nM T59604 C9TY3J 44446157 IC50 = 450 nM T59604 C7ZNF8 44446175 IC50 = 800 nM T59604 C6J4VA 44446177 EC50 = 32 nM T59604 C19UPX 44446178 EC50 = 88 nM T59604 CYE3V6 44446187 EC50 = 75 nM T59604 C5TF6G 44446188 EC50 = 1580 nM T59604 CRHA84 44446189 EC50 = 24 nM T59604 C9WB8K 44446190 EC50 = 24 nM T59604 CHQI08 44447839 EC50 = 0.42 nM T59604 C57ZXB 44447840 EC50 = 1.6 nM T59604 CN7P0S 44447841 EC50 = 0.61 nM T59604 CF7ED5 44447842 EC50 = 6.75 nM T59604 C3V1TO 44447843 EC50 = 0.72 nM T59604 CB4YK8 44447844 EC50 = 1.79 nM T59604 C9LCW5 44447845 EC50 = 34 nM T59604 CHW3R7 44447846 EC50 = 3.1 nM T59604 C5XNV0 44447848 EC50 = 33.2 nM T59604 C24VRW 44447850 EC50 = 1.26 nM T59604 C87OWH 44447852 EC50 = 0.51 nM T59604 C5RFG7 44447853 EC50 = 1.11 nM T59604 CBF75I 44447854 EC50 = 1.66 nM T59604 C5PNS2 44447855 EC50 = 0.34 nM T59604 CK1QX4 44447856 EC50 = 1.04 nM T59604 C4ZC3O 44447857 EC50 = 0.45 nM T59604 CUT47D 44449864 EC50 = 3 nM T59604 CZU9Y0 44449891 EC50 = 0.9 nM T59604 C13VTX 44449922 EC50 = 2.9 nM T59604 C1AQ4F 44449923 EC50 = 105 nM T59604 CC0FR8 44449924 EC50 = 521 nM T59604 C0V8JF 44449955 EC50 = 0.2 nM T59604 CIX4J9 44449956 EC50 = 3.1 nM T59604 C0O9SE 44449987 EC50 = 0.2 nM T59604 C3NQW9 44449988 EC50 = 0.7 nM T59604 CA67EK 44450015 EC50 = 1.3 nM T59604 C40TMA 44450016 EC50 = 0.6 nM T59604 C5XJE2 44450017 EC50 = 1.8 nM T59604 CKP79S 44450044 EC50 = 40 nM T59604 CN0C2P 44450045 EC50 = 27 nM T59604 CG5FL6 44450046 EC50 = 3.3 nM T59604 C0SD3B 44450070 EC50 = 204 nM T59604 C6S8YR 44450071 EC50 = 140 nM T59604 CCUH90 44450100 EC50 = 8.4 nM T59604 C9JZX1 44450101 EC50 = 0.64 nM T59604 C4SCA9 44450102 EC50 = 11 nM T59604 C3DG5S 44450103 EC50 = 4.1 nM T59604 CM3LC9 44450104 EC50 = 1.4 nM T59604 C0LOA1 44450105 EC50 = 33 nM T59604 CU1I0E 44450132 EC50 = 4.4 nM T59604 C61EIS 44450133 EC50 = 14.7 nM T59604 C9Y4QK 44450134 EC50 = 32 nM T59604 CF4WP5 44450135 EC50 = 23 nM T59604 C0H1PK 44450137 EC50 = 70 nM T59604 C45JKU 44450169 EC50 = 26 nM T59604 CL5I7Z 44452749 EC50 = 0.3981 nM T59604 C8EX9A 44452750 EC50 = 1.995 nM T59604 CV52TF 44452776 EC50 = 125.89 nM T59604 C6C9KF 44452777 EC50 = 39.81 nM T59604 C8R3DW 44452778 EC50 = 794.33 nM T59604 CX4RI1 44452806 EC50 = 100 nM T59604 C6N7KC 44452825 EC50 = 39.81 nM T59604 CXJ24Q 44452826 EC50 = 39.81 nM T59604 CIF7L4 44452827 EC50 = 630.96 nM T59604 CM3SB0 44452885 EC50 = 100 nM T59604 CTY80L 44452887 EC50 = 158.49 nM T59604 CWNM19 44452929 EC50 = 19.95 nM T59604 CCZF71 44452932 EC50 = 1.995 nM T59604 C6M5SL 44453070 EC50 = 316.23 nM T59604 CN54QX 44453097 EC50 = 316.23 nM T59604 CZL3X4 44453123 EC50 = 0.5012 nM T59604 CV13SO 44454060 EC50 = 0.8 nM T59604 C56TGO 44454092 EC50 = 19 nM T59604 C8L7PU 44454117 EC50 = 0.5 nM T59604 CZ6K7I 44454302 EC50 = 23 nM T59604 CPM4W2 44454303 EC50 = 0.3 nM T59604 C3O4BS 44454304 EC50 = 19 nM T59604 C83YHV 44454337 EC50 = 0.4 nM T59604 C30CSY 44454338 EC50 = 19 nM T59604 CZ21VY 44454367 EC50 = 0.6 nM T59604 C46EKP 44454368 EC50 = 302 nM T59604 CTJ75W 44454397 EC50 = 2470 nM T59604 C2B4SN 44454398 EC50 = 27 nM T59604 C1PGK4 44454399 EC50 = 22 nM T59604 CDF7M8 44454432 EC50 = 150 nM T59604 CSX29M 44560945 EC50 = 0.9 nM T59604 C5QLC6 44570698 EC50 = 19.95 nM T59604 CHD4F5 44570699 EC50 = 3.981 nM T59604 C9KD1J 44570700 EC50 = 1.995 nM T59604 CX86AU 44570702 EC50 = 2.512 nM T59604 CQ5X3W 44570761 EC50 = 31.62 nM T59604 C2Z3HJ 44570762 EC50 = 316.23 nM T59604 C4D0AV 44570763 EC50 = 1 nM T59604 C17ONP 44570764 EC50 = 0.3162 nM T59604 C84LHN 44570765 EC50 = 0.3981 nM T59604 CE15GU 44570920 EC50 = 7.943 nM T59604 CWF7R1 44570921 EC50 = 15.85 nM T59604 C61CHS 44570922 EC50 = 398.11 nM T59604 CPAI69 44570923 EC50 = 31.62 nM T59604 CTN23G 44570960 EC50 = 0.2512 nM T59604 CP46TB 44570961 EC50 = 3.162 nM T59604 C53BQS 44570962 EC50 = 0.05012 nM T59604 C9ZW2M 44570963 EC50 = 0.1585 nM T59604 C37FQE 44570964 EC50 = 15.85 nM T59604 CUZ8G1 44570965 EC50 = 1.259 nM T59604 C5HZ8J 44570966 EC50 = 0.5012 nM T59604 CG58BJ 44570967 EC50 = 5.012 nM T59604 CKS86A 44571002 EC50 = 0.1995 nM T59604 C2B7WE 44571003 EC50 = 6.31 nM T59604 C3AWE9 44571004 EC50 = 10 nM T59604 CJB06H 44571005 EC50 = 7.943 nM T59604 C6JB2C 44576254 IC50 > 1000 nM T59604 C5TF9Y 44576256 IC50 = 0.25 nM T59604 CD3T1I 44577060 Ki = 240 nM T59604 CVS6Q8 44579640 EC50 = 4000 nM T59604 C6D3LJ 44579641 EC50 = 2000 nM T59604 CCY9F0 44579643 EC50 = 90 nM T59604 C2ZJM0 44579686 EC50 = 4000 nM T59604 CHY2F7 44579752 EC50 = 14000 nM T59604 CVH40U 44579753 EC50 > 10000 nM T59604 C5AHW3 44579754 EC50 > 10000 nM T59604 CDT3M9 44579755 EC50 = 900 nM T59604 CC8AI0 44579756 EC50 = 7 nM T59604 C0MH7I 44579774 EC50 >= 10 nM T59604 C4WN7B 44579775 EC50 = 40 nM T59604 C87QLB 44579776 EC50 = 80 nM T59604 CE9U6O 44579777 EC50 = 150 nM T59604 C2YS5Q 44579778 EC50 = 50 nM T59604 CPM02Q 44579801 EC50 = 220 nM T59604 C5U4QZ 44579802 EC50 = 10 nM T59604 CC5PZ6 44579803 EC50 = 260 nM T59604 CNH16J 44579804 EC50 = 60 nM T59604 C4HIN8 44579805 EC50 = 20 nM T59604 CG2JM1 44579821 EC50 = 140 nM T59604 CY5V2L 44579822 EC50 = 90 nM T59604 C7P8JA 44579823 EC50 = 3 nM T59604 C15AZN 44579824 EC50 = 120 nM T59604 CERM69 44579840 EC50 = 20 nM T59604 CKB1J3 44579841 EC50 = 30 nM T59604 CO3J8L 44579842 EC50 = 1260 nM T59604 CA7W8Q 44579843 EC50 = 90 nM T59604 C34IHS 44579844 EC50 >= 10 nM T59604 C4CA5O 44579857 EC50 = 200 nM T59604 CDE7M9 44579858 EC50 = 50 nM T59604 CNM2G5 44579859 EC50 >= 10 nM T59604 C69CYU 44579860 EC50 = 250 nM T59604 CB79UF 44579861 EC50 = 120 nM T59604 CAG89V 44579879 EC50 = 140 nM T59604 C78VMJ 44579880 EC50 = 30 nM T59604 CB01KP 44579881 EC50 = 780 nM T59604 CT2H0M 44579882 EC50 = 40 nM T59604 C4Y5HF 44579883 EC50 = 120 nM T59604 C7NZY6 44579906 EC50 = 1200 nM T59604 C6C1JT 44579907 EC50 = 20 nM T59604 CLR28I 44579908 EC50 = 1500 nM T59604 C6NB2S 44579909 EC50 = 180 nM T59604 CL7VA5 44579919 EC50 = 2000 nM T59604 CH85UT 44579958 EC50 = 1000 nM T59604 CD5KM4 44579959 EC50 = 600 nM T59604 CNZ5W9 44579995 EC50 > 10000 nM T59604 CBTA01 44579996 EC50 = 2000 nM T59604 CGN8D7 44579998 EC50 > 10000 nM T59604 C4L7TJ 44580028 EC50 = 5000 nM T59604 C79IVU 44580029 EC50 > 10000 nM T59604 CXJY26 44580030 EC50 = 440 nM T59604 C9Q5LO 44580031 EC50 = 330 nM T59604 CMX14O 44580032 EC50 = 9000 nM T59604 C4AMJ8 44582533 IC50 = 55000 nM T59604 C7KBO6 44582534 IC50 = 889000 nM T59604 CQI0D4 45102707 EC50 > 10000 nM T59604 CSEP-69 45102708 EC50 > 1000 nM T59604 C7FSM2 46865987 IC50 = 12.2 nM T59604 CTEA12 46880461 IC50 = 25 nM T59604 CK8A1O 46880462 IC50 = 12 nM T59604 C9KDP4 46880463 IC50 = 640 nM T59604 CEQ6V4 46880495 IC50 = 280 nM T59604 CISM52 46880496 IC50 = 68 nM T59604 C8ZSM3 46880497 IC50 = 6500 nM T59604 CODR73 46880498 IC50 = 46.5 nM T59604 CHJ5Y6 46880566 IC50 = 77 nM T59604 CE9PG2 46880567 IC50 = 147 nM T59604 C01PGO 46880568 IC50 = 6 nM T59604 CS7L4X 46880569 IC50 = 26 nM T59604 C0PXY7 46880628 IC50 = 9.1 nM T59604 CD37LU 46880629 IC50 = 2.1 nM T59604 CUY89F 46880630 IC50 = 4.1 nM T59604 C4P6XS 46880631 IC50 = 2.9 nM T59604 CJ53KF 46880672 IC50 = 7 nM T59604 CYJC08 46880673 IC50 = 136 nM T59604 C1RI9O 46880674 IC50 = 64 nM T59604 CJ5LO0 46880675 IC50 = 17.7 nM T59604 COT5L9 46880724 IC50 = 14.3 nM T59604 C8TW5J 46880725 IC50 = 9 nM T59604 CMUZ29 46880726 IC50 = 20 nM T59604 CMS56Q 46880727 IC50 = 13 nM T59604 CA1V5O 46880770 IC50 = 37.2 nM T59604 CE1OL2 46880771 IC50 = 33.7 nM T59604 CEXW19 46880772 IC50 = 12.7 nM T59604 CE57JN 46880773 IC50 = 42.2 nM T59604 CT1S6C 46880811 IC50 = 143 nM T59604 C6OX9Z 46880812 IC50 = 65 nM T59604 CB1VX9 46880813 IC50 = 244.6 nM T59604 C6CS2B 46880814 IC50 = 123 nM T59604 C6PCS9 46880844 IC50 = 338.7 nM T59604 CJOU53 46880845 IC50 = 42 nM T59604 C2EFB5 46880846 IC50 = 31 nM T59604 C0LJP6 46882103 IC50 = 108 nM T59604 CX1KS6 46882104 IC50 = 310 nM T59604 CB67WR 46882105 IC50 = 444 nM T59604 CH5T9E 46882106 IC50 = 625 nM T59604 CR2C3J 46882152 IC50 = 429 nM T59604 C3KSB8 46882153 IC50 = 682 nM T59604 C39QLM 46882154 IC50 = 5615 nM T59604 C2QM9K 46882155 IC50 = 1649 nM T59604 C43CSF 46882156 IC50 = 846 nM T59604 CE9Z1W 46882196 IC50 = 474 nM T59604 CJ9GQ6 46882197 IC50 = 241 nM T59604 CA18GZ 46882198 IC50 = 97 nM T59604 C6OY8D 46882199 IC50 = 263 nM T59604 C0AU3L 46882236 IC50 = 128 nM T59604 CNZI39 46882237 IC50 = 138 nM T59604 C4YUO1 46882238 IC50 = 161 nM T59604 CGTQ20 46882239 IC50 = 69 nM T59604 CMEL41 46882270 IC50 = 77 nM T59604 CFL3C6 46882271 IC50 = 14 nM T59604 CAVT63 46882272 IC50 = 8 nM T59604 C0IF2Y 46882273 IC50 = 28 nM T59604 CIGP20 46882302 EC50 > 1000 nM T59604 CJG6E9 46882303 EC50 > 1000 nM T59604 CW2Z0V 46882305 IC50 = 16 nM T59604 C9IDW2 46882306 IC50 = 21 nM T59604 C20XKF 46882307 IC50 = 2 nM T59604 C69AMR 46882349 EC50 > 10000 nM T59604 CFZV45 46882350 EC50 > 1000 nM T59604 CSF43I 46882393 EC50 > 1000 nM T59604 CB3QV6 46882394 EC50 = 3.981 nM T59604 C01GKH 46882395 EC50 = 3.981 nM T59604 CX7D3V 46882396 EC50 = 19.95 nM T59604 C4BH9E 46882458 EC50 = 79.43 nM T59604 CJ69NR 46882460 EC50 > 1000 nM T59604 C3FA8G 46882519 EC50 > 10000 nM T59604 CF8IJ2 46882520 EC50 = 79.43 nM T59604 CQN87I 46882521 EC50 = 1584.89 nM T59604 C56ULO 46882522 EC50 = 158.49 nM T59604 CRZ95W 46882582 EC50 = 630.96 nM T59604 CX72IN 46882583 EC50 > 10000 nM T59604 CHS14B 46882671 EC50 > 1000 nM T59604 C2OU8F 46882673 EC50 > 10000 nM T59604 CP84OR 46882710 EC50 > 10000 nM T59604 CPFM68 46882711 EC50 > 10000 nM T59604 CC05XO 46882712 EC50 > 10000 nM T59604 CL3EI9 46882713 EC50 > 10000 nM T59604 CZ15LN 46882714 EC50 > 1000 nM T59604 CD24US 46882752 EC50 > 1000 nM T59604 CAN69D 46882753 EC50 > 1000 nM T59604 C0RQA4 46882754 EC50 > 1000 nM T59604 CBXT24 46882756 EC50 > 1000 nM T59604 C4DLJ2 46882763 IC50 = 40 nM T59604 CH6G4Q 46882766 IC50 = 272 nM T59604 C39WEJ 46882794 EC50 > 1000 nM T59604 CTJ41Q 46882795 EC50 > 1000 nM T59604 C4OZ1U 46882796 EC50 > 1000 nM T59604 CDK0Q3 46882797 EC50 > 1000 nM T59604 CMC4E5 46882804 IC50 = 46 nM T59604 CCUI47 46882805 IC50 = 30 nM T59604 C3NSG9 46882807 IC50 = 1715 nM T59604 C4OQ6D 53248756 Ki = 22 nM T59604 C28QUB 53373577 Ki = 3.311 nM T59604 CC8Q1D 53390181 IC50 = 12.59 nM T59604 CV0P1K 53390538 IC50 = 30.2 nM T59604 CZ0WI6 53391301 IC50 = 37.15 nM T59604 C7XZ1I 54458823 EC50 = 3 nM T59604 CP1W5M 56926173 EC50 = 68 nM T59604 C30RQU 56926461 Ki = 6 nM T59604 C9IEJ8 56942098 IC50 = 4 nM T59604 C6AZ3E 56942099 Ki = 8 nM T59604 CCF90X 56942242 Ki = 0.8 nM T59604 C2AT0L 56942243 Ki = 2 nM T59604 C7ZF9T 56942244 Ki = 12 nM T59604 CX3L9I 56942385 Ki = 46 nM T59604 CVE3F7 56942387 IC50 = 43 nM T59604 CO9KV2 56942388 Ki = 17 nM T59604 CM7PW5 56942535 Ki = 46 nM T59604 CW4QD9 57345597 Ki = 2 nM T59604 CBQK82 57345598 Ki = 3.1 nM T59604 C3REK0 57345599 Ki = 0.2 nM T59604 CX49PE 57345600 Ki = 0.16 nM T59604 CI9UT0 57391292 Ki = 3.1 nM T59604 CH67TI 57391293 Ki = 0.4 nM T59604 C78LTO 57391294 Ki = 3.4 nM T59604 CGB71E 57393073 Ki = 0.1 nM T59604 CRE41N 57394797 Ki = 6.6 nM T59604 CS41PI 57394881 Ki = 0.05 nM T59604 C3D4AH 57394882 Ki = 5 nM T59604 CKDZ14 57398339 Ki = 0.9 nM T59604 CSA36Q 57398340 Ki = 0.01 nM T59604 CE5JQ8 57398341 Ki = 0.2 nM T59604 C7NE4P 57398342 Ki = 0.26 nM T59604 C8Y4UJ 57398343 Ki = 1.9 nM T59604 C8CG2S 57399248 Ki = 1 nM T59604 C18OVS 57400002 Ki = 0.01 nM T59604 CJO70A 57400003 Ki = 2.6 nM T59604 CL2IT5 57401797 Ki = 1.7 nM T59604 CKA34L 57401798 Ki = 6.7 nM T59604 CM15JF 57401799 Ki = 0.3 nM T59604 CGS82D 57401800 Ki = 0.5 nM T59604 CF0CA4 57401801 Ki = 0.6 nM T59604 C53DGY 57401802 Ki = 1.5 nM T59604 C8VI1X 57401803 Ki = 0.27 nM T59604 CX6JR2 57422673 IC50 = 23 nM T59604 CD40CR 57422686 IC50 = 0.15 nM T59604 CRI4K2 57422687 IC50 = 0.29 nM T59604 C6JZ4C 57422688 IC50 = 0.67 nM T59604 CR8S3Q 57422690 IC50 = 0.53 nM T59604 CYSA42 57422692 IC50 = 0.33 nM T59604 CO85NH 57422695 IC50 = 3.9 nM T59604 CTS3E6 57422696 IC50 = 15 nM T59604 CW92IZ 57422697 IC50 = 120 nM T59604 C43BGV 57422730 IC50 = 13 nM T59604 CO1KA7 57422749 IC50 = 65 nM T59604 C2IO0J 57422760 IC50 = 8.7 nM T59604 CSF86Y 57422761 IC50 = 8.6 nM T59604 CJO7S5 57422768 IC50 = 0.48 nM T59604 C03XVS 57422776 IC50 = 5.1 nM T59604 CK1BZ0 57422789 IC50 = 1.3 nM T59604 C59DSI 57422791 IC50 = 8.8 nM T59604 CKMP13 57422792 IC50 = 0.31 nM T59604 CBY54J 57422793 IC50 = 0.62 nM T59604 C2U1VH 57422817 IC50 = 0.77 nM T59604 CH9ZJ5 57785733 IC50 = 0.69 nM T59604 C39VTY 57785737 IC50 = 4.2 nM T59604 CY3NF5 57797614 IC50 = 11 nM T59604 CZ6Q9X 57797640 IC50 = 2 nM T59604 C54DIC 58438451 Ki = 10.47 nM T59604 CPI4W9 58438460 Ki = 12.88 nM T59604 C9UK7P 58438475 Ki = 6.31 nM T59604 CBCA81 58438487 Ki = 9.12 nM T59604 C1FM5N 59446099 IC50 > 10000 nM T59604 CV52YE 59446101 IC50 = 1200 nM T59604 C0V5UB 59446102 IC50 > 10000 nM T59604 C9S1IF 59446103 IC50 > 10000 nM T59604 CS92LO 59446104 IC50 > 10000 nM T59604 C3KB2O 59446107 IC50 = 1340 nM T59604 CQE13H 59446108 IC50 > 10000 nM T59604 C8PKR2 59446111 IC50 > 10000 nM T59604 CS3JD0 59446113 IC50 > 10000 nM T59604 CRJ38P 59446116 IC50 = 51000 nM T59604 C0INX9 59446117 IC50 > 10000 nM T59604 CL50PI 59446120 IC50 = 771 nM T59604 C2G6QX 59446121 IC50 > 10000 nM T59604 CHZQ39 59446122 IC50 > 10000 nM T59604 C3OG9S 59446123 IC50 > 10000 nM T59604 CHNR24 59446125 IC50 > 10000 nM T59604 CP07SK 59446126 IC50 > 10000 nM T59604 CZIC40 59446128 IC50 > 10000 nM T59604 CA0W9Q 59446130 IC50 = 19500 nM T59604 C6QMA8 59446134 IC50 > 10000 nM T59604 CX5Y1T 59446135 IC50 = 808 nM T59604 C7OCA4 59446138 IC50 = 723 nM T59604 CU03SE 59446139 IC50 = 11200 nM T59604 CRQB10 59446141 IC50 = 3740 nM T59604 C29SIX 59446142 IC50 > 10000 nM T59604 CA03QR 59446143 IC50 = 45000 nM T59604 C7IPK4 59446145 IC50 = 568 nM T59604 CU17OY 59446146 IC50 > 10000 nM T59604 CTYL12 59446149 IC50 > 10000 nM T59604 C7OB4H 59446150 IC50 = 3250 nM T59604 CP42MS 59446154 IC50 = 8170 nM T59604 CLV4J8 60165265 IC50 = 38 nM T59604 CYH80K 60194838 IC50 > 10000 nM T59604 CD8S1Q 60194839 IC50 > 10000 nM T59604 CG28AQ 60195018 IC50 = 3860 nM T59604 C5CXK6 60195019 IC50 = 3610 nM T59604 C2GWS0 60195020 IC50 = 5410 nM T59604 C9QK5Y 60195112 IC50 = 1170 nM T59604 CZ7MK5 60195113 IC50 = 4550 nM T59604 CV6XG5 60195114 IC50 = 85600 nM T59604 C45OTP 60195115 IC50 > 10000 nM T59604 CP4RF0 60195284 IC50 = 16100 nM T59604 CW51MB 60195285 IC50 = 465 nM T59604 CX7M6C 60195286 IC50 = 729 nM T59604 CXQ0J6 60195379 IC50 = 1640 nM T59604 C2FPA0 60195645 IC50 > 10000 nM T59604 C4NEG2 60195731 IC50 > 10000 nM T59604 C2YO0F 66601728 IC50 = 7 nM T59604 CT9B1S 66788278 IC50 = 2 nM T59604 C78XLS 66813470 IC50 = 200 nM T59604 C4UP0J 67405379 Ki = 3.981 nM T59604 C7M8VC 67406334 Ki = 4.571 nM T59604 CPV39L 67406727 Ki = 9.2 nM T59604 CU32ZC 67407161 Ki = 15.49 nM T59604 C3GSR6 67407808 Ki = 9.12 nM T59604 CWY79V 67408128 Ki = 7.413 nM T59604 C3BHE6 67410074 Ki = 15.49 nM T59604 C8LM1Q 67457995 EC50 = 0.6 nM T59604 CM3PW8 70681018 IC50 = 3 nM T59604 CMDT94 70681019 IC50 = 79 nM T59604 CY0IK4 70681020 IC50 = 196 nM T59604 C87FCB 70681021 IC50 = 2.5 nM T59604 C5D2MP 70681022 IC50 = 16.5 nM T59604 CN4G3U 70681025 IC50 > 10000 nM T59604 C3J9KZ 70682036 Ki = 14 nM T59604 CKSP64 70682037 IC50 = 4.6 nM T59604 C16WKZ 70683143 IC50 = 28 nM T59604 CHPA96 70683144 IC50 > 10000 nM T59604 CAKY84 70683149 IC50 = 50 nM T59604 CD5TR3 70684154 IC50 = 231 nM T59604 C79PIV 70684155 Ki = 27 nM T59604 C97XVQ 70685218 IC50 = 171 nM T59604 C4O8XG 70685219 IC50 = 4.1 nM T59604 CK8A6W 70685225 IC50 = 3 nM T59604 C1P4OY 70686292 IC50 = 25 nM T59604 CJ2UM8 70686293 Ki = 14 nM T59604 C8RP9Q 70687379 IC50 = 143 nM T59604 CL1WU4 70687380 IC50 = 8 nM T59604 C5QG9Y 70687383 IC50 = 6 nM T59604 CS0HG6 70688404 IC50 = 211 nM T59604 CN7RS4 70689440 IC50 = 7 nM T59604 CGRS90 70689441 IC50 = 20 nM T59604 CCI32L 70690449 Ki = 20 nM T59604 C1AC0G 70691550 IC50 = 0.2 nM T59604 CF8I9T 70691551 IC50 = 1 nM T59604 C8ZI6D 70691552 IC50 = 2.5 nM T59604 C27NFD 70692600 Ki = 14 nM T59604 C8ST6F 70692601 Ki = 11 nM T59604 COI36G 70692602 Ki = 114 nM T59604 CKSH84 70692603 Ki = 25 nM T59604 CM3T7V 70693640 IC50 = 26 nM T59604 CH8GC3 70693641 IC50 = 12 nM T59604 C5LQ9B 70693643 IC50 > 10000 nM T59604 CB4F0R 70693644 IC50 = 7 nM T59604 CG5QA4 70694647 IC50 = 2980 nM T59604 CLK3G6 70694648 Ki = 52 nM T59604 CBX49P 70694649 Ki = 23 nM T59604 C93XHS 70695747 Ki = 4.4 nM T59604 CG0QY5 70695748 IC50 = 314 nM T59604 C62ZQG 70695749 IC50 = 313 nM T59604 CAH70F 70696687 Ki = 152 nM T59604 CI62QY 70696688 Ki = 17 nM T59604 C94JEF 70696689 Ki = 206 nM T59604 CK2T6G 71449740 IC50 = 220 nM T59604 CC6Z0B 71449752 IC50 > 10000 nM T59604 CXZ4K1 71449753 IC50 = 2540 nM T59604 C4BT1J 71449838 EC50 = 168.6 nM T59604 CHNV45 71449843 EC50 > 1000 nM T59604 CZBF56 71451551 IC50 = 129 nM T59604 C7A5LH 71451563 IC50 = 24 nM T59604 CSQF84 71451564 IC50 = 251 nM T59604 CL8V0U 71451652 EC50 > 1000 nM T59604 C0IBC7 71452183 Ki = 100 nM T59604 CN08XO 71453389 IC50 > 10000 nM T59604 CWK3J2 71453390 IC50 = 38 nM T59604 C1XR4A 71453391 IC50 = 25 nM T59604 CTIF57 71453392 IC50 = 110 nM T59604 CY7CZ1 71453404 IC50 = 47 nM T59604 C5KO6D 71453405 IC50 = 700 nM T59604 CTME20 71453485 EC50 = 624.4 nM T59604 CR2F8D 71453488 EC50 = 6.7 nM T59604 C7WR4T 71453489 EC50 = 2.8 nM T59604 C5J9NH 71455085 IC50 = 64 nM T59604 CURV69 71455104 IC50 > 10000 nM T59604 C7IX2J 71455105 IC50 = 140 nM T59604 CK3OR6 71455106 IC50 = 525 nM T59604 CU8BM9 71455196 EC50 > 1000 nM T59604 C5GBY7 71455197 EC50 = 9.4 nM T59604 CBN67Z 71456897 IC50 = 1 nM T59604 CD2RP7 71456910 IC50 = 110 nM T59604 CU30QE 71456984 EC50 = 183.7 nM T59604 CD3X1J 71456992 EC50 = 5.7 nM T59604 C39NDE 71458746 IC50 = 1160 nM T59604 COF8H7 71458747 IC50 = 213 nM T59604 CUJ34O 71458847 Ki = 31.3 nM T59604 CH8UP0 71458848 EC50 = 240.9 nM T59604 C2REN0 71458849 Ki = 22.1 nM T59604 C5FG2U 71458850 EC50 = 96.8 nM T59604 CHT38B 71458859 EC50 = 13.1 nM T59604 CFT7E2 71460564 IC50 = 1470 nM T59604 CEW73V 71460565 IC50 = 1180 nM T59604 CY3R0Z 71460566 IC50 > 10000 nM T59604 CW7EY5 71460576 IC50 = 1390 nM T59604 CDXZ12 71460577 IC50 = 273 nM T59604 CU6M4L 71460578 IC50 = 111 nM T59604 C3OLW2 71460658 Ki = 34.9 nM T59604 C1OPU6 71460659 EC50 = 2.1 nM T59604 CCV93Y 71460664 EC50 = 119.6 nM T59604 CT79JP 71460665 EC50 = 498.1 nM T59604 CVJY40 71462272 IC50 = 239 nM T59604 C1UQO9 71462273 IC50 = 47 nM T59604 C8Q0SD 71462274 IC50 = 2780 nM T59604 CE7J5X 71462275 IC50 > 10000 nM T59604 COLZ61 71462276 IC50 > 10000 nM T59604 C9W5VI 71462373 EC50 > 1000 nM T59604 CEO4H0 71462380 EC50 = 124.1 nM T59604 CK7Z6F 71462381 EC50 = 17.9 nM T59604 C6Y4WM 71462382 EC50 = 161.3 nM T59604 CE2BA8 71716660 EC50 = 0.7943 nM T59604 CEX25Q 72190449 Ki = 275.42 nM T59604 C79XFZ 72190450 IC50 = 1096.48 nM T59604 C7NYG0 72190451 Ki = 25.12 nM T59604 C6PE7F 72190452 Ki = 1380.38 nM T59604 CN4D2K 72191050 Ki = 27.54 nM T59604 CL1A6K 72191051 Ki = 16.22 nM T59604 C4J7PB 73346226 Ki = 3630.78 nM T59604 CUR4F2 73346227 Ki < 20892.96 nM T59604 C2B1GF 73347725 IC50 = 15.85 nM T59604 CCI07X 73350118 IC50 = 12 nM T59604 CBX06Q 73350846 Ki = 25118.86 nM T59604 C2TK7H 73352329 Ki = 1122.02 nM T59604 C93IHF 73352330 Ki < 29512.09 nM T59604 CL8T4U 73355325 Ki = 1698.24 nM T59604 CD63YS 73356869 Ki < 30199.52 nM T59604 CB4Y7R 89768546 IC50 = 6500 nM T59604 C4OP6C 90644553 Ki = 10.47 nM T59604 CF0MJ8 90644554 Ki = 69.18 nM T59604 CG4E8W 90665845 IC50 = 0.12 nM T59604 C1S7YU 90665846 IC50 = 1.5 nM T59604 C8B1RN 90665847 IC50 = 0.28 nM T59604 CCQ67W 90665848 IC50 = 16 nM T59604 C2DF8V 90665849 IC50 = 59 nM T59604 CGB7U8 90665850 IC50 = 1.1 nM T59604 C67YNO 90665851 IC50 = 1.1 nM T59604 C2E6NI 90665852 IC50 = 12 nM T59604 C97PUB 90666011 IC50 = 7.3 nM T59604 CU9OP3 90666012 IC50 = 1.6 nM T59604 C8O2ZM 90666013 IC50 = 1.8 nM T59604 C3ND7I 90666014 IC50 = 32 nM T59604 CSJE46 90666015 IC50 = 44 nM T59604 CN31ZU 90666016 IC50 = 4000 nM T59604 C6W4GH 90666017 EC50 = 1.3 nM T59604 C0D5FT 90666018 IC50 = 6.1 nM T59604 CMX8H0 90666019 IC50 = 370 nM T59604 CK8V1H 90666020 IC50 = 23 nM T59604 CTY8Q0 90666021 IC50 = 7.6 nM T59604 CF03DJ 90666022 IC50 = 120 nM T59604 C2O3UE 90666023 IC50 = 15 nM T59604 C4AP0G 90666024 IC50 = 5.1 nM T59604 CV3J8C 90666025 IC50 = 5 nM T59604 CD48KA 90666026 IC50 = 40 nM T59604 C7EIY6 90666027 IC50 = 1.7 nM T59604 C89PMV 90666028 IC50 = 120 nM T59604 CM2H6G 90666029 IC50 = 2.7 nM T59604 C9G5KP 90666030 IC50 = 5.7 nM T59604 C6NIZ9 90666031 IC50 = 1.6 nM T59604 CPVX39 90666032 IC50 = 12 nM T59604 C0U5BY 90666033 IC50 = 200 nM T59604 C45OBZ 90666034 IC50 = 60 nM T59604 C5WQN4 90666035 IC50 = 980 nM T59604 C85AMH 90666036 IC50 = 500 nM T59604 CKF14A 90666037 IC50 = 190 nM T59604 CM7ED5 90666038 IC50 = 52 nM T59604 CU2T3C 90666039 IC50 = 0.91 nM T59604 C59YXE 90666040 IC50 = 4.8 nM T59604 C6QZL4 90666041 IC50 = 11 nM T59604 CY35OV 90666042 IC50 = 27 nM T59604 C0V5EC 91826086 IC50 > 30000 nM T59604 CXV5R4 118709470 IC50 = 210 nM T59604 CE08TK 118709471 IC50 = 76 nM T59604 CK21QD 118709472 IC50 = 4700 nM T59604 C9ECO8 118709473 IC50 > 10000 nM T59604 C4P0SO 118709502 IC50 = 0.24 nM T59604 CI6FA2 118709503 IC50 = 0.57 nM T59604 CYK5M2 118709504 IC50 = 33 nM T59604 C70QKY 118709505 IC50 = 0.92 nM T59604 CCDV59 118709506 IC50 = 0.4 nM T59604 CT87MK 118709507 IC50 = 7.2 nM T59604 C80ORL 118718706 EC50 = 440 nM T59604 CFP2D9 118722878 IC50 = 6.31 nM T59604 CY9MF7 118725954 Ki = 49 nM T59604 C1W9RO 118725955 Ki > 50 nM T59604 C0T8AU 118725956 Ki = 6.4 nM T59604 C76QKE 118725957 Ki > 50 nM T59604 CPY60A 118725958 Ki = 166 nM T59604 CN21JF 118725959 Ki > 50 nM T59604 C4C2OQ 118725960 Ki = 13 nM T59604 C9LG8K 118725961 Ki = 4 nM T59604 C6KD7W 118725962 Ki = 263 nM T59604 CKQT19 118725963 Ki = 127 nM T59604 CAQ80I 118725964 Ki = 139 nM T59604 C2QS3P 118725965 Ki = 20 nM T59604 CSFY18 118725966 Ki = 28 nM T59604 CR2NZ9 122178176 EC50 = 6 nM T59604 C1Q0GC 122178177 EC50 = 189.2 nM T59604 CT5QV3 122178178 EC50 = 63.1 nM T59604 CK3W1J 122178179 EC50 = 29 nM T59604 CJ3YC7 122178180 EC50 = 60.2 nM T59604 C0DKP8 122178182 EC50 > 1000 nM T59604 C92LNJ 122178184 EC50 = 316.23 nM T59604 CKJ1U0 122178185 EC50 = 251.19 nM T59604 C3LKE9 122178186 EC50 = 99.9 nM T59604 CE0WR2 122178187 IC50 = 77.62 nM T59604 C4XDU8 122178188 EC50 = 39.81 nM T59604 C5Q7WR 122178189 IC50 = 70.79 nM T59604 CZV5P9 122178599 IC50 > 1000 nM T59604 CJ8CE4 122178600 IC50 = 122 nM T59604 C7YJ1F 122178601 IC50 = 88 nM T59604 CW3M9R 122178602 IC50 = 193 nM T59604 CU2I3P 122178603 IC50 = 130 nM T59604 CU48DB 122178604 IC50 = 380 nM T59604 CKWJ12 122178605 IC50 = 8.8 nM T59604 C6FN0V 122178606 IC50 = 2.1 nM T59604 C1HG6X 122178607 IC50 = 4.6 nM T59604 CTF3L2 122178608 IC50 = 3.4 nM T59604 CL31JE 122178609 IC50 = 2 nM T59604 CTIU14 122178610 IC50 = 6 nM T59604 C4A8XV 122178611 IC50 = 108 nM T59604 C1UB6L 122178612 IC50 = 79 nM T59604 C1GY8B 122178613 IC50 = 65 nM T59604 CLB32A 122178614 IC50 = 230 nM T59604 CIO35B 122178615 IC50 = 82 nM T59604 CJS9X1 122178616 IC50 = 100 nM T59604 CCH92O 122180014 IC50 = 84 nM T59604 CZ1C2A 122180015 IC50 = 150 nM T59604 C84EGT 122180016 IC50 = 260 nM T59604 CH4CF5 122180017 IC50 = 11 nM T59604 C9C6OK 122180018 IC50 = 36 nM T59604 CJ7OV3 122180019 IC50 = 180 nM T59604 C2E3MQ 122180020 IC50 = 24 nM T59604 CFG0I3 122180021 IC50 = 6.9 nM T59604 CA9P7Z 122180022 IC50 = 47 nM T59604 C0GD4B 122180023 IC50 = 7.2 nM T59604 CC7TK9 122180024 IC50 = 5.4 nM T59604 CRN0L6 122180025 IC50 = 42 nM T59604 C3HU8Z 122180026 IC50 = 0.96 nM T59604 CNZ3M0 122180027 IC50 = 0.23 nM T59604 CK49AE 122182043 IC50 = 0.39 nM T59604 CT0R6V 122182046 IC50 = 0.42 nM T59604 C7RLI5 122182047 IC50 = 0.3 nM T59604 CY8DA3 122182189 IC50 = 3 nM T59604 CBHG71 122182190 IC50 = 0.44 nM T59604 C87ASV 127045651 Ki > 1000 nM T59604 CAL12J 127045834 Ki > 1000 nM T59604 C2A3GB 127045858 IC50 = 3 nM T59604 CHPL37 127045859 Ki = 3 nM T59604 COK5L4 127046472 EC50 = 70 nM T59604 CO4A9F 127046473 Ki = 8 nM T59604 C36DRS 127046806 Ki = 154 nM T59604 C1MOG4 127046807 Ki = 62 nM T59604 CKQ0Y6 127046808 Ki > 1000 nM T59604 CHSJ34 127046956 IC50 = 2 nM T59604 C80BUK 127046957 IC50 = 4 nM T59604 CXT70M 127047362 IC50 = 130 nM T59604 CD42FM 127047363 Ki > 1000 nM T59604 C06JWX 127047409 EC50 = 170 nM T59604 CAO45B 127047523 Ki = 3 nM T59604 CZA7Y9 127047525 EC50 = 0.8 nM T59604 C27NXH 127047654 Ki = 62 nM T59604 C51JYG 127047655 IC50 = 7 nM T59604 C1C3JS 127048038 IC50 = 115 nM T59604 C26YTW 127048059 Ki = 2.5 nM T59604 C3JDM0 127048060 Ki = 17 nM T59604 C2TGW6 127048061 EC50 = 82 nM T59604 CZ2RL1 145948708 Ki = 50 nM T59604 C2OCP4 145948725 Ki = 2 nM T59604 C27NUT 145949381 EC50 = 25 nM T59604 C54ACE 145949595 EC50 = 19.95 nM T59604 CAB18Y 145949755 EC50 = 12.59 nM T59604 C6P9QW 145949880 IC50 = 501.19 nM T59604 C91DXZ 145950201 IC50 = 63.1 nM T59604 C8N5JL 145950261 EC50 = 125.89 nM T59604 C76GPL 145950336 EC50 = 0.1 nM T59604 CMP8T0 145950877 EC50 = 23 nM T59604 C6LXA0 145950963 EC50 = 158.49 nM T59604 CU81XO 145950987 EC50 = 50.12 nM T59604 C3YMF2 145951150 EC50 = 3 nM T59604 CAF83G 145952396 EC50 = 158.49 nM T59604 C0JZA8 145952404 EC50 = 251.19 nM T59604 C30MRB 145952740 EC50 = 15 nM T59604 C8QJW2 145953016 EC50 = 19 nM T59604 CHG09C 145953855 EC50 = 31.62 nM T59604 C25NVO 145954311 IC50 = 1260 nM T59604 CAW62C 145955250 EC50 = 125.89 nM T59604 C90KIG 145955718 EC50 = 251.19 nM T59604 CZ7IP5 145956026 EC50 = 5 nM T59604 C1J0BV 145956061 EC50 = 1.259 nM T59604 C9K4AQ 145956415 EC50 = 250 nM T59604 CR9DQ8 145956659 EC50 = 47 nM T59604 CFG2A0 145956753 EC50 = 236 nM T59604 CQVJ40 145957075 EC50 = 2.512 nM T59604 CU80KI 145957404 EC50 = 125.89 nM T59604 CASL75 145957443 IC50 = 184 nM T59604 CFZJ34 145957574 EC50 = 1.585 nM T59604 CG40FJ 145958317 EC50 = 25.12 nM T59604 CF0V3H 145958487 EC50 = 7 nM T59604 CWT43A 145958774 EC50 = 226 nM T59604 C4DMP9 145959007 EC50 = 39.81 nM T59604 CY75UJ 145959787 EC50 = 36 nM T59604 C03WXR 145961213 EC50 = 19.95 nM T59604 CF7GE0 145962494 EC50 = 10 nM T59604 CEY3A6 145974293 EC50 = 19.95 nM T59604 CN70VQ 145975725 EC50 > 7700 nM T59604 CWO02C 145979268 EC50 = 439 nM T59604 C3XBR0 145979819 EC50 = 484 nM T59604 C3QNO0 145980333 EC50 = 298 nM T59604 CV85ZH 145980382 EC50 = 29.4 nM T59604 C35FBK 145981196 EC50 = 483 nM T59604 C06LYT 145981343 EC50 = 2164 nM T59604 CD5NG2 145981687 EC50 = 40.7 nM T59604 CNIJ28 145981794 EC50 = 67 nM T59604 C9XC3S 145982096 IC50 > 30000 nM T59604 CM2HZ8 145982683 EC50 > 30000 nM T59604 C06VYC 145984632 EC50 = 363 nM T59604 CB0LX5 145986080 EC50 = 73 nM T59604 C8M9ZU 145986461 EC50 = 1276 nM T59604 CIL85G 145986870 EC50 = 85.7 nM T59604 CA6OW1 145987684 IC50 = 192 nM T59604 CYKQ65 145988286 EC50 = 70 nM T59604 CB4IN0 145988557 EC50 = 117 nM T59604 CXU4N1 145988582 IC50 = 2005 nM T59604 CJ5K7A 145988647 EC50 = 634 nM T59604 CRM2K5 145988894 EC50 = 51 nM T59604 CQ2N4K 145989762 EC50 > 30000 nM T59604 CG78YI 145989916 IC50 = 1300 nM T59604 CJ38OD 145990051 IC50 = 2367 nM T59604 CU3H4A 145990956 IC50 = 919 nM T59604 C58ETM 145991389 IC50 = 2330 nM T59604 C3PVM4 145991797 IC50 = 4010 nM T59604 CPX20Q 145991822 IC50 = 1130 nM T59604 C1DZK8 145991945 EC50 = 937 nM T59604 C7K8NJ 145992125 EC50 = 121 nM T59604 CD2V3K 145992142 EC50 = 189 nM T59604 CT57AZ 145992253 EC50 = 96 nM T59604 C6GEP2 145992835 EC50 = 84.8 nM T59604 CI4VH0 145992854 IC50 = 148 nM T59604 C3I8LB 145993313 EC50 = 970 nM T59604 CB2T3U 145993528 EC50 = 10.6 nM T59604 C15OAH 145993628 IC50 = 106 nM T59604 C02SLN 145993758 IC50 = 1510 nM T59604 C7ZU8A 145994050 EC50 = 194 nM T59604 CEP45Z 145994299 IC50 = 2700 nM T59604 C1PY8C 155526063 Ki = 3.4 nM T59604 C9JM2W 155529391 Ki = 2.7 nM T59604 CLQ4R5 155537651 Ki = 3.05 nM T59604 CAV10C 155540883 Ki = 1.26 nM T59604 C15KZH 155551597 Ki = 6.45 nM T59604 C2W8HU 155557019 EC50 = 2.5 nM T59604 CG7X4P 155561671 Ki = 55 nM T59604 CXC5Q2 46905972 EC50 = 3 nM T59604 D01LKO 44576255 IC50 = 540 nM T59604 D02NZI 9890863 IC50 = 4 nM T59604 D07JZB 44576248 IC50 = 12 nM T59604 D07QLZ 44576252 IC50 = 14 nM T59604 D08GTH 10190715 IC50 = 530 nM T59604 D09QPV 44576253 IC50 = 120 nM T59604 D0C3OY 25091011 Ki = 76.7 nM T59604 D0G8TL 44576249 IC50 = 58 nM T59604 D0J2YB 23631116 Ki = 4 nM T59604 D0L3AP 44576251 IC50 = 60 nM T59604 D0L3EP 25124566 IC50 = 3.981 nM T59604 D0PQ7A 44576250 IC50 = 210 nM T59604 D0U2QP 46882764 IC50 = 4300 nM T59604 D0XR6A 44576247 IC50 = 2.6 nM T59604 D0ZG7W 11441554 IC50 = 7 nM T94255 C8CUS5 1295523 IC50 = 400 nM T94255 CW59YI 2264067 IC50 = 1500 nM T94255 C4WI8K 2950887 IC50 = 1600 nM T94255 CEK6B1 139300630 IC50 > 10000 nM T94255 C4S7LQ 155514237 IC50 = 1300 nM T94255 C7X1EI 155519256 IC50 = 2800 nM T94255 CRO0K3 155530772 IC50 = 5900 nM T94255 C3C9GI 155535515 IC50 = 4700 nM T94255 CG23CH 155556141 IC50 = 4900 nM T94255 CY1JZ0 155564517 IC50 = 3600 nM T94255 D0G2MU 10229 IC50 = 29000 nM T67272 D0RA5Q 72172 IC50 = 0.81 ug.mL-1 T67272 D0U2JP 4369359 IC50 > 100000 nM T67272 D07SDQ 969516 IC50 = 15500 nM T67272 D0F2JS 15547703 IC50 = 680 nM T67272 D0T2IQ 443600 IC50 = 0.32 ug.mL-1 T67272 CKN1L3 20479 Ki = 10000 nM T67272 C0V9WL 73324 IC50 > 100 ug.mL-1 T67272 C8X2GZ 76808 IC50 = 1000000 nM T67272 CG48YC 97710 Ki = 27500 nM T67272 CP1JX4 124031 IC50 = 15 ug.mL-1 T67272 CKWA31 125415 Ki = 17000 nM T67272 C01SOJ 130013 Ki = 19 nM T67272 C2QHX5 182612 Ki = 53000 nM T67272 C6JM7L 182750 IC50 = 30 ug.mL-1 T67272 CV0J8H 182751 IC50 = 41.7 ug.mL-1 T67272 CGT6C5 276114 IC50 = 93.7 ug.mL-1 T67272 C7FP6H 277936 IC50 = 800000 nM T67272 CDBF98 281242 Ki = 10600 nM T67272 CNM0P3 391527 IC50 = 101400 nM T67272 CW10CK 439518 Ki = 200 nM T67272 CESM72 439530 IC50 = 41000 nM T67272 C5RO7V 469541 IC50 = 20 nM T67272 C0TYO2 477693 IC50 = 10.3 ug.mL-1 T67272 C7G3CT 477696 IC50 > 100 ug.mL-1 T67272 C4TRL6 721814 IC50 > 100 ug.mL-1 T67272 CO3KZ2 741570 IC50 = 84.7 ug.mL-1 T67272 CE28KQ 850934 IC50 = 6.7 ug.mL-1 T67272 C0L7TD 1235479 IC50 = 5.4 ug.mL-1 T67272 C6L1VE 1551321 Ki = 167 nM T67272 C2HQJ7 2302144 IC50 = 29.5 ug.mL-1 T67272 C3MR8Q 2817201 Ki = 2010 nM T67272 C59OKR 4330464 IC50 = 12400 nM T67272 CY36MH 4369380 Ki > 10000 nM T67272 CK8VJ3 5311145 Ki = 430000 nM T67272 CAQP85 5713154 Ki = 5950 nM T67272 C7AZE5 6930803 IC50 = 38400 nM T67272 CYQ8J7 9849506 IC50 = 28 nM T67272 C2DMP6 9861924 IC50 = 3.5 ug.mL-1 T67272 CFMG63 9886974 IC50 = 11.4 ug.mL-1 T67272 C30OXI 9990739 Ki = 3850 nM T67272 C5Q6BJ 9995375 IC50 > 100 ug.mL-1 T67272 CYH3C6 10061400 IC50 = 17.8 ug.mL-1 T67272 CV7SK8 10064801 IC50 = 309200 nM T67272 CWU9N2 10198228 IC50 > 100 ug.mL-1 T67272 C27AJQ 10245523 IC50 = 1000000 nM T67272 C0JD8Z 10333136 IC50 = 29 ug.mL-1 T67272 CTZQ69 10347030 IC50 = 1345 nM T67272 CK8T4C 10381531 IC50 = 4.3 ug.mL-1 T67272 C79UAO 10381586 IC50 > 100 ug.mL-1 T67272 C6GWB8 10401570 IC50 = 0.9 ug.mL-1 T67272 CL3H9I 10491923 IC50 = 16 ug.mL-1 T67272 CJ2RK6 10492044 IC50 = 70.7 ug.mL-1 T67272 C3YS4K 10659346 IC50 = 49.5 ug.mL-1 T67272 CN5KG9 10661540 IC50 = 9.6 ug.mL-1 T67272 C1LSP2 10779050 IC50 > 100 ug.mL-1 T67272 CD2GP9 10784566 IC50 > 100 ug.mL-1 T67272 C04XQH 10850290 IC50 = 54.3 ug.mL-1 T67272 C3ODA7 10945796 Ki = 1015 nM T67272 CN5H0B 10970861 Ki = 7.2 nM T67272 C5OPG0 11127644 Ki = 0.79 nM T67272 C10KPB 11142955 Ki = 2 nM T67272 CIOY84 11723708 IC50 = 15 ug.mL-1 T67272 CI2OP1 11942810 IC50 = 122500 nM T67272 CO0W1G 12749378 IC50 = 500000 nM T67272 C7RI2M 13168364 IC50 = 20 nM T67272 C29UOD 13226135 IC50 = 310000 nM T67272 CC9DK6 13384604 IC50 = 30400 nM T67272 CCX02R 13491256 IC50 = 25 nM T67272 C9F5CM 13491267 IC50 = 40 nM T67272 CF19DX 13509139 Ki = 341 nM T67272 CYV1F7 13784835 IC50 > 100 ug.mL-1 T67272 CP8L5J 14104451 IC50 = 38600 nM T67272 C94FPE 14434173 IC50 = 44.1 ug.mL-1 T67272 CT3L5Q 14542146 Ki = 660000 nM T67272 CP4OT8 14542149 Ki = 79000 nM T67272 CC17MK 15078261 Ki = 20 nM T67272 CW9ER1 15159715 IC50 = 30 nM T67272 CWNE58 15159721 IC50 = 21 nM T67272 CO1F2B 15342195 IC50 = 1000000 nM T67272 CE1P6J 15719279 Ki = 2500 nM T67272 CD28WR 15719282 Ki = 10500 nM T67272 CYR87Z 15719283 Ki = 18000 nM T67272 C4Y1HP 15849848 Ki = 7420 nM T67272 CB6WK0 16121107 Ki = 80000 nM T67272 CZQ8O9 16121199 Ki = 100000 nM T67272 CT01PQ 16739331 IC50 > 100000 nM T67272 C7YJZ5 17748252 IC50 = 3100 nM T67272 C9J8IN 18445902 IC50 = 53800 nM T67272 CYR08N 19366756 Ki = 8 nM T67272 C7GDU9 20038035 IC50 > 100 ug.mL-1 T67272 CF4VL0 21120524 Ki = 120 nM T67272 C8JSI4 23628284 IC50 > 100000 nM T67272 CFP01R 24828743 Ki = 100 nM T67272 C9LUM1 24828881 Ki = 27.54 nM T67272 CY9W8O 24860300 IC50 > 100000 nM T67272 C1CMY7 24884567 IC50 = 1800 nM T67272 C0VL7B 24890303 Ki = 52.48 nM T67272 C4R6BZ 24901452 Ki = 500 nM T67272 CTJU08 24975348 Ki = 1000 nM T67272 CIO26D 25022463 IC50 = 48500 nM T67272 CYZ2J7 25141282 IC50 = 21700 nM T67272 CP0YF8 25146956 IC50 = 81800 nM T67272 C12AVL 25146957 IC50 = 71300 nM T67272 C10MBE 25146958 IC50 = 24100 nM T67272 CIUY75 25146959 IC50 = 68400 nM T67272 C5MG9N 25146960 IC50 = 149300 nM T67272 C83IOD 25147056 IC50 = 74800 nM T67272 C1IA0W 25147057 IC50 = 135300 nM T67272 CB3W1I 25147058 IC50 = 161800 nM T67272 CC35MZ 25147059 IC50 = 196400 nM T67272 CO5H9V 25147060 IC50 = 232700 nM T67272 CM20ZC 25147061 IC50 = 29800 nM T67272 C2KZ0T 25147062 IC50 = 62200 nM T67272 C5RMI2 25147153 IC50 = 98400 nM T67272 C43YCQ 25147154 IC50 = 51400 nM T67272 CPQW89 25147155 IC50 = 121500 nM T67272 CQ3I6B 25147156 IC50 = 46600 nM T67272 C2LHR1 25147157 IC50 = 70600 nM T67272 CA34UT 25147158 IC50 = 121700 nM T67272 C3R0DB 25147159 IC50 = 72300 nM T67272 CV4ZE9 25147248 IC50 = 82600 nM T67272 C73HYI 25147249 IC50 = 137300 nM T67272 CV14TY 25147250 IC50 = 33500 nM T67272 CUW8X2 25147251 IC50 = 56100 nM T67272 C0Z7NX 25147252 IC50 = 96600 nM T67272 CU1KO6 25147352 IC50 = 78400 nM T67272 C7RS3Y 25195667 IC50 = 8000 nM T67272 C7IHC9 44207184 IC50 = 120000 nM T67272 C12CDQ 44254309 Ki = 512.86 nM T67272 C8EI1G 44254310 Ki = 181.97 nM T67272 CD3L0N 44254402 Ki = 8.511 nM T67272 CHT0Z1 44254404 Ki = 218.78 nM T67272 CW7LB9 44254495 Ki = 50.12 nM T67272 C5FDC2 44254496 Ki = 12.59 nM T67272 CR01EW 44256381 IC50 = 800 nM T67272 CUBV96 44276209 Ki = 4500 nM T67272 C34DUK 44276215 Ki = 2300 nM T67272 C9CUN1 44276216 Ki = 1900 nM T67272 C0Q1WI 44276218 IC50 = 75000 nM T67272 C32JVB 44276289 Ki = 45000 nM T67272 C79TMD 44276303 Ki = 210 nM T67272 C4JB1Z 44276401 Ki = 25000 nM T67272 CQX6J3 44276410 Ki = 35 nM T67272 CV5MC9 44276625 Ki = 7300 nM T67272 CHP16B 44276842 Ki = 2700 nM T67272 CQP05Z 44283812 IC50 = 1000000 nM T67272 C52KDH 44283814 IC50 = 1000000 nM T67272 CZT7Y3 44283829 IC50 = 3400 nM T67272 CUOI41 44283840 IC50 = 5000 nM T67272 CJ72SM 44283849 IC50 = 1000000 nM T67272 C36NHS 44283851 IC50 = 1000000 nM T67272 CK6ZW2 44283857 IC50 = 3800 nM T67272 C3PQR5 44283863 IC50 = 1000000 nM T67272 C0UG6P 44283886 IC50 = 1000000 nM T67272 C1YQM9 44283908 IC50 = 85000 nM T67272 CZG67T 44283924 IC50 = 146000 nM T67272 CE4NA8 44283925 IC50 = 2900 nM T67272 CT0O3D 44284085 IC50 = 783000 nM T67272 C6SFV4 44284086 IC50 = 1000000 nM T67272 CN9A8Q 44284101 IC50 = 2400 nM T67272 C7K8JV 44323547 IC50 = 1628 nM T67272 CRAI45 44323558 IC50 = 28000 nM T67272 CW2GK4 44344567 Ki = 11 nM T67272 CS75VD 44360285 Ki = 24000 nM T67272 C4QON9 44368427 IC50 = 10.2 ug.mL-1 T67272 C8FB1S 44368725 IC50 = 38.2 ug.mL-1 T67272 CE83AK 44368726 IC50 > 100 ug.mL-1 T67272 CW9BG0 44368735 IC50 > 100 ug.mL-1 T67272 C37TIM 44368736 IC50 = 40.5 ug.mL-1 T67272 C1U4IX 44458314 IC50 = 20 nM T67272 CRTB46 44458322 IC50 = 20 nM T67272 C5XS9L 44481133 IC50 = 23700 nM T67272 C3PYH7 44481390 IC50 = 64300 nM T67272 C38HFR 44481392 IC50 = 28800 nM T67272 CRC8F9 44481394 IC50 = 30800 nM T67272 CPJI36 44481396 IC50 = 23300 nM T67272 C9SG6K 44481398 IC50 = 38100 nM T67272 C0G2AC 44481400 IC50 = 18900 nM T67272 CFI01J 44481402 IC50 = 42000 nM T67272 CZ4KP3 44481661 IC50 = 16900 nM T67272 C3B9EX 44481663 IC50 = 41000 nM T67272 CO5D8W 44481665 IC50 = 21500 nM T67272 CY3KS0 44481667 IC50 = 15800 nM T67272 CXRA28 44481669 IC50 = 22100 nM T67272 C0M5WT 44481671 IC50 = 16600 nM T67272 C1EGD7 44481673 IC50 = 11300 nM T67272 CC5NV2 44481931 IC50 = 15400 nM T67272 CY5QH7 44481933 IC50 = 16900 nM T67272 CDCT90 44481935 IC50 = 9400 nM T67272 CQUL08 44481937 IC50 = 10900 nM T67272 CVM9E2 44481939 IC50 = 12500 nM T67272 C01YEO 44481941 IC50 = 5300 nM T67272 CJD57G 44481943 IC50 = 9200 nM T67272 C7JK5B 44482208 IC50 = 32100 nM T67272 CH3B9V 44482210 IC50 = 20700 nM T67272 CMQA93 44482214 IC50 = 13200 nM T67272 CRZ9P0 44482218 IC50 = 9700 nM T67272 CZ4H7R 44560401 Ki = 5000 nM T67272 C70AIZ 44560402 Ki = 55000 nM T67272 C63VWA 44560403 Ki = 49000 nM T67272 CRX2G5 44560404 Ki = 17000 nM T67272 CA4IF6 44560405 Ki = 11000 nM T67272 C57LTE 44560406 Ki = 10000 nM T67272 C2F3TI 44560407 Ki = 16000 nM T67272 CC3GY2 44560408 Ki = 20000 nM T67272 C9YE7J 44560409 Ki = 21000 nM T67272 C1OEW5 44560410 Ki = 17000 nM T67272 CU4G1S 44560411 Ki = 13000 nM T67272 C2Y0OT 44560412 Ki > 100000 nM T67272 CG7BQ8 44560457 Ki = 33000 nM T67272 C1RK3C 44560557 Ki > 100000 nM T67272 C42VEQ 44560558 Ki = 69000 nM T67272 C0J6LB 44563970 IC50 = 73700 nM T67272 C3US0I 44569010 IC50 = 24800 nM T67272 C3TAN1 44569011 IC50 = 51200 nM T67272 CF0L2W 44569012 IC50 = 74600 nM T67272 CGI35S 44569013 IC50 = 41400 nM T67272 C8PO5Q 44569024 IC50 = 168600 nM T67272 C52JXP 44569036 IC50 = 43800 nM T67272 CU1NI6 44569037 IC50 = 36400 nM T67272 CS9CH4 44569038 IC50 = 61300 nM T67272 C63ZQK 44569039 IC50 = 47300 nM T67272 C2WE7H 44569040 IC50 = 39500 nM T67272 CO8FB4 44569058 IC50 = 134700 nM T67272 C3K4ED 44569059 IC50 = 53600 nM T67272 CPWR76 44569060 IC50 = 47500 nM T67272 CU39FK 44569061 IC50 = 68900 nM T67272 CR6H0X 44569062 IC50 = 28400 nM T67272 CTWR37 44569063 IC50 = 31600 nM T67272 C6M9SH 44569081 IC50 = 114300 nM T67272 C5RN7U 44569082 IC50 = 33500 nM T67272 CQ9OA7 44569083 IC50 = 26300 nM T67272 CCV74H 44576563 IC50 = 54900 nM T67272 C59TCG 44576564 IC50 = 75800 nM T67272 CMI9S4 44576565 IC50 = 92600 nM T67272 CD8ZI4 44576587 IC50 = 155800 nM T67272 CQ87CS 44576614 IC50 = 173700 nM T67272 CJY2W3 44576615 IC50 = 124300 nM T67272 CL92CH 44576616 IC50 = 150600 nM T67272 CIU84E 44576617 IC50 = 168100 nM T67272 C9ODS1 44576618 IC50 = 134800 nM T67272 C35DWL 44576631 IC50 = 61800 nM T67272 C6ZL1U 44576632 IC50 = 73200 nM T67272 CK09LV 44576633 IC50 = 57800 nM T67272 CFL76T 44576634 IC50 = 82700 nM T67272 CC58GQ 44576635 IC50 = 106700 nM T67272 CZNQ90 44593458 IC50 = 141900 nM T67272 CR3Q4N 44593532 IC50 = 41600 nM T67272 CTWL91 46193025 IC50 = 7300 nM T67272 CMLG10 46882676 Ki = 128.82 nM T67272 CTO1Q8 46882677 Ki = 54.95 nM T67272 C19YDM 46886333 Ki = 53000 nM T67272 C9HPU0 46886351 Ki = 27500 nM T67272 CHE51J 49795928 IC50 = 83000 nM T67272 CS1TY7 49795932 IC50 = 104000 nM T67272 CP9WB0 49840768 Ki = 3588 nM T67272 C51YRX 49840770 Ki = 11100 nM T67272 CJ3Z7V 49840772 Ki = 16800 nM T67272 CS3I8G 49840774 Ki = 7245 nM T67272 C3IT5V 49840844 Ki = 10800 nM T67272 CYBW37 49840846 Ki = 48900 nM T67272 CFEC23 49840848 Ki = 9217 nM T67272 C64XMG 49840850 Ki = 5436 nM T67272 CNU1Q7 49840921 Ki = 11900 nM T67272 C7S9QA 50913428 IC50 = 3000 nM T67272 CO4XE9 50913573 IC50 = 5100 nM T67272 CQ90FE 52941108 Ki = 57000 nM T67272 CU4HK1 52943524 Ki = 5974 nM T67272 C9HRG4 52946764 Ki = 50000 nM T67272 C89EGH 52947188 Ki = 841 nM T67272 CU58OG 53257413 Ki = 4955 nM T67272 C6XY5R 53259047 Ki = 1074 nM T67272 C7AXD8 53259048 Ki = 5413 nM T67272 CX51OK 53259216 Ki = 1571 nM T67272 CBS92H 53259217 Ki = 12000 nM T67272 C8RZW7 53259219 Ki > 100000 nM T67272 C4KZ7R 53259403 Ki > 100000 nM T67272 CA0Q2E 53259404 Ki > 100000 nM T67272 C6FU2G 53259405 Ki > 100000 nM T67272 CLSC37 53261358 Ki = 12000 nM T67272 CXMC12 53261359 Ki = 3283 nM T67272 C3Q4ZR 53261360 Ki = 8345 nM T67272 C48JHC 53320960 IC50 > 1000000 nM T67272 C9QWK0 53322291 IC50 = 300000 nM T67272 CO0X3H 53324937 Ki = 20000 nM T67272 CGP68U 53324939 Ki = 60000 nM T67272 CN12AO 53353383 IC50 > 100000 nM T67272 C51GUC 53354365 IC50 > 100000 nM T67272 CRJ5P9 53354369 IC50 > 100000 nM T67272 C4G2HT 53354470 IC50 > 100000 nM T67272 CFS7N9 53494936 Ki = 11 nM T67272 CN53IO 53792079 Ki = 691 nM T67272 CGF98A 54585162 Ki = 1299 nM T67272 CLP2C1 54753981 IC50 = 32690 nM T67272 CGTV56 56658262 IC50 = 248350 nM T67272 CV46HL 56665195 IC50 = 289950 nM T67272 C3L5SO 56665196 IC50 = 615560 nM T67272 CH4M6V 56665197 IC50 = 66340 nM T67272 CSU81T 56672275 IC50 = 39430 nM T67272 CF75JN 56953635 IC50 = 30000 nM T67272 CQ64IE 56953636 IC50 > 100000 nM T67272 C9RJF3 56953637 IC50 = 500 nM T67272 CM7VP3 56953638 IC50 > 70000 nM T67272 C1BWY5 56953762 IC50 = 54000 nM T67272 C4VJI0 56953763 IC50 = 45000 nM T67272 C7JYZ1 56953764 IC50 = 30000 nM T67272 CH67KO 56953765 IC50 > 100000 nM T67272 CSW96U 56955172 IC50 = 44000 nM T67272 CFG17Q 56955173 IC50 = 65000 nM T67272 C76MEC 56955271 IC50 > 100000 nM T67272 CWGA37 56955272 IC50 = 13500 nM T67272 C28VDY 56955273 IC50 = 500 nM T67272 C1QSV9 56955274 IC50 = 48000 nM T67272 C1T2QI 60144811 IC50 = 420 nM T67272 CI4AV6 70073083 IC50 = 9600 nM T67272 C64XBZ 70681347 IC50 = 37000 nM T67272 C4N3VW 70681348 IC50 > 70000 nM T67272 C5EHM1 70681503 IC50 > 100000 nM T67272 CFP12D 70683616 IC50 = 75000 nM T67272 CYVJ36 70683617 IC50 = 122000 nM T67272 CYD34L 70685541 IC50 = 65000 nM T67272 C1DZ3J 70685542 IC50 = 47000 nM T67272 C4BN0J 70689859 IC50 = 10000 nM T67272 CB4ZL3 70690154 IC50 = 39000 nM T67272 CHM4W5 70692015 IC50 = 64000 nM T67272 CJ3OY4 70692312 IC50 = 22000 nM T67272 C0HFX4 70694371 IC50 = 16000 nM T67272 CFT06N 70696054 IC50 > 70000 nM T67272 C6MW3C 70696243 IC50 = 27000 nM T67272 C2IAG5 70696244 IC50 > 100000 nM T67272 CLE79H 70696450 IC50 = 110000 nM T67272 CA6IB0 71450469 IC50 = 910 nM T67272 CT5J7F 71452300 IC50 = 790 nM T67272 C23NVO 71452301 IC50 = 6900 nM T67272 CU3KE8 71453804 Ki = 1000 nM T67272 C5K8WS 71454094 IC50 = 940 nM T67272 CP2D3C 71454095 IC50 = 1100 nM T67272 C3VQW4 71455829 IC50 = 6400 nM T67272 CKR4D0 71459517 IC50 = 1500 nM T67272 C6UQW4 71461261 IC50 = 3000 nM T67272 C9QE5X 71462985 IC50 = 480 nM T67272 CL0P1Y 71584425 IC50 = 1310 nM T67272 C1BF6E 71584426 IC50 = 530 nM T67272 CMRA35 71584427 IC50 = 610 nM T67272 C6STG3 71584428 IC50 = 700 nM T67272 C42XYH 71584672 IC50 = 650 nM T67272 C2TYL8 71584673 IC50 = 730 nM T67272 CS3T9Q 71602397 IC50 = 3120 nM T67272 CIWZ87 71602398 IC50 = 15160 nM T67272 CJK3H7 71603240 IC50 = 9580 nM T67272 CMJF12 71603241 IC50 = 16190 nM T67272 CY7M2C 71603243 IC50 = 10940 nM T67272 C4M9AB 71603244 IC50 = 97490 nM T67272 C9ZJ2B 71603245 IC50 = 19660 nM T67272 C5OB3M 73348808 IC50 = 12100 nM T67272 C28UIX 73356287 IC50 = 793000 nM T67272 CEM9F5 73672383 IC50 = 65290 nM T67272 CRU02V 74766022 Ki = 0.23 nM T67272 C05HWU 86140993 Ki = 1660 nM T67272 CF35LZ 87495845 Ki = 41100 nM T67272 CUD73A 90645555 Ki > 10000 nM T67272 C0YOU8 90664312 IC50 = 9400 nM T67272 CDQF80 90664420 IC50 = 14100 nM T67272 CYND40 90672013 IC50 = 1100 nM T67272 CG9N2T 90672014 IC50 = 420 nM T67272 C34ALI 94005078 IC50 = 220 nM T67272 C8BNV9 95566324 Ki = 19 nM T67272 CX29SF 97550302 Ki = 19 nM T67272 CDA72U 101882336 Ki = 0.21 nM T67272 CVS60Z 118720629 Ki = 4.8 nM T67272 C4VWL9 118720630 Ki = 2.4 nM T67272 C71CKB 118720631 Ki = 146 nM T67272 CCQ74S 118720632 Ki = 24.2 nM T67272 C8JDP5 118720633 Ki = 1.7 nM T67272 CE9X4G 118720634 Ki = 2.1 nM T67272 CW87DK 118720635 Ki = 1.3 nM T67272 CKIF61 118720636 Ki = 27.8 nM T67272 CJ6MY3 118720637 Ki = 2.1 nM T67272 CP5V7M 118720638 Ki = 0.69 nM T67272 CQ6K5N 118720639 Ki = 1.1 nM T67272 CWL1M3 122195270 IC50 = 85000 nM T67272 CN6UZ5 122195271 IC50 = 20000 nM T67272 C6CV7K 122195272 IC50 > 70000 nM T67272 CHE75Z 122195273 IC50 > 70000 nM T67272 C6RY2A 122195274 IC50 = 22000 nM T67272 C14TSF 122195275 IC50 = 62000 nM T67272 CIE12T 122195276 IC50 = 32000 nM T67272 C4DXT1 122195277 IC50 = 52000 nM T67272 CNV2J7 122195278 IC50 > 100000 nM T67272 C8C0HD 124196349 Ki = 172 nM T67272 CLSB73 124196351 Ki = 497 nM T67272 C7IK1U 124196354 Ki = 71.2 nM T67272 CPU97K 124196355 Ki = 49.1 nM T67272 CUE28O 124196356 Ki = 40 nM T67272 C4FV5U 124196371 Ki = 348 nM T67272 C9Y8LQ 124196373 Ki = 29.1 nM T67272 CWVI53 124196382 Ki = 560 nM T67272 CG46VB 124196383 Ki = 188 nM T67272 C0Z5QW 124196384 Ki = 82.1 nM T67272 CGEJ47 124196385 Ki = 37.3 nM T67272 C8Z1BF 124196387 Ki = 300 nM T67272 C9MPY5 127025893 IC50 = 120 nM T67272 C3TF8V 127037842 IC50 = 280 nM T67272 CUO5V9 127039573 Ki = 118 nM T67272 CM0VT4 127048200 Ki = 37700 nM T67272 CTL4Z8 127048201 Ki = 499 nM T67272 CBQ4S3 127048202 Ki = 275 nM T67272 CC96VU 127048834 Ki = 782 nM T67272 CRCB36 127048872 Ki = 2510 nM T67272 CTY5D4 127049157 Ki = 6040 nM T67272 CF3HO2 127049196 Ki = 13500 nM T67272 C03XKF 127049491 Ki = 391 nM T67272 CFW6M1 127049492 Ki = 5740 nM T67272 CL6D0Z 127049497 Ki = 4450 nM T67272 C4I1RH 127049824 Ki = 397 nM T67272 C2A1MZ 127050130 Ki = 1220 nM T67272 CA4MP3 127050430 Ki = 1110 nM T67272 CJT5R9 127050433 Ki = 3220 nM T67272 C0N2LE 127050745 Ki = 2550 nM T67272 C9GBD2 127051304 Ki = 1490 nM T67272 CLK50R 127051701 Ki = 207 nM T67272 C2BUZ7 127051959 Ki = 357 nM T67272 CK81ME 127051999 Ki = 78 nM T67272 CAC25R 127052273 Ki = 297 nM T67272 C3FMN7 127052612 Ki = 2890 nM T67272 CHA9Q6 127052870 Ki = 65 nM T67272 CJM96B 127053163 Ki = 3290 nM T67272 CLJ9F6 145949706 IC50 = 3200 nM T67272 C25EDJ 145952430 IC50 = 1950 nM T67272 C32LGX 145952863 IC50 = 740 nM T67272 C0MC6U 145955648 IC50 = 870 nM T67272 CQNE67 145956257 IC50 = 270 nM T67272 CN84MC 145956662 IC50 = 5370 nM T67272 CN1CQ3 145957783 IC50 = 1680 nM T67272 CB03UD 145960195 IC50 = 5600 nM T67272 CM2D9J 145961321 IC50 = 6500 nM T67272 CK5P6I 145961499 IC50 = 4800 nM T67272 C4J0HA 145963210 IC50 = 5000 nM T67272 C27HIP 145963359 IC50 = 6900 nM T67272 CZU0S1 145963748 IC50 = 280 nM T67272 CL1DE4 145965106 IC50 = 10200 nM T67272 C38IXU 145966119 IC50 = 190 nM T67272 CP9ZD1 145971617 Ki = 80 nM T67272 C1VOU2 145976275 Ki = 1010 nM T67272 CM7YB8 145998092 Ki = 4.5 nM T67272 CSF69J 155511374 Ki = 131 nM T67272 C3WTA6 155513618 Ki > 1000000 nM T67272 CKZ21H 155513922 Ki = 205 nM T67272 CX2ZT9 155513964 Ki = 604 nM T67272 CF7LE9 155514400 Ki = 442 nM T67272 C8GB3J 155514541 Ki = 277 nM T67272 CUGK20 155515062 Ki = 102 nM T67272 C6LCH3 155515796 Ki = 430 nM T67272 CT2C5J 155517371 Ki = 704 nM T67272 CIGF73 155517640 Ki = 19.2 nM T67272 C4AE5F 155518479 Ki = 978 nM T67272 CA3TM6 155518679 Ki = 111 nM T67272 CG2RF3 155520398 Ki = 8.2 nM T67272 CM1ES6 155523825 Ki = 745 nM T67272 CNF48I 155525687 IC50 = 810 nM T67272 C6G0MI 155528995 Ki = 163 nM T67272 CZ2BF0 155529155 Ki = 185 nM T67272 CI2P4Z 155533156 Ki = 235 nM T67272 C7HJ5U 155534393 IC50 = 620 nM T67272 CZN50A 155535841 IC50 = 990 nM T67272 C8C1EI 155540506 IC50 = 3300 nM T67272 C56KWP 155543532 IC50 = 650 nM T67272 CY02VQ 155546277 Ki = 462 nM T67272 CX1CW7 155547815 Ki = 240 nM T67272 C5I9HJ 155548213 Ki = 158 nM T67272 CH61FB 155550504 Ki = 23.4 nM T67272 CA08LZ 155550520 Ki = 522 nM T67272 CWM3Q7 155550895 Ki = 182 nM T67272 C71FAU 155553065 Ki = 43.1 nM T67272 CK3Q4N 155556136 Ki = 137 nM T67272 CHY95K 155559649 Ki = 366 nM T67272 CRQ4V7 155559773 Ki = 170 nM T67272 CM43NT 155559807 Ki = 4420 nM T67272 C9S2FL 155562411 Ki = 919 nM T67272 C07NIE 155563089 Ki = 119 nM T67272 CMUF64 155565532 Ki = 175 nM T67272 C6J9LE 155567025 Ki = 631 nM T67272 C5UH8A 155567330 Ki = 138 nM T67272 CEO6S0 155568852 Ki = 156 nM T67272 C0VK3G 44344579 Ki = 4.8 nM T67272 C2PVI1 44344594 Ki = 2.9 nM T67272 CHEX85 445715 Ki = 2.62 nM T67272 D04DTE 53259050 Ki = 240 nM T67272 D04QJY 123982 Ki = 7000 nM T67272 D06AFP 11436221 IC50 = 3400 nM T67272 D0A7GO 44309732 Ki = 20000 nM T67272 D0H5BG 53494934 Ki = 0.06 nM T67272 D0I6RL 11723962 IC50 > 100000 nM T67272 D0L3PY 123814 Ki = 56.23 nM T59045 D0R3QY 5665 Ki = 850000 nM T59045 D00BRD 126 IC50 = 4.1 ug.mL-1 T59045 D09SWE 31244 IC50 > 1000000 nM T59045 D0B5YS 1183 IC50 = 17100 nM T59045 D0NH9P 135 IC50 > 1000000 nM T59045 D0X7BT 125 IC50 > 1000000 nM T59045 CY8P0F 227 IC50 > 5000000 nM T59045 C6X9CB 978 IC50 > 1000000 nM T59045 C0F1EW 6271 IC50 = 176000 nM T59045 CLE87P 7419 IC50 > 5000000 nM T59045 CV9N2M 7469 IC50 = 188000 nM T59045 CR0U3Y 115067 IC50 > 1000000 nM T59045 CSJ7V0 277942 IC50 > 5000000 nM T59045 C97XKM 506073 IC50 > 5000000 nM T59045 CR3OI1 571807 IC50 > 5000000 nM T59045 CA6EQ4 1514158 IC50 > 5000000 nM T59045 C4Q6ZR 3000722 Ki = 91000 nM T59045 C7EP1S 7016465 Ki = 13000000 nM T59045 CDY5C8 10011990 Ki = 100000 nM T59045 CHX1O3 10103265 Ki = 125000 nM T59045 CFH15U 10419269 Ki = 2300000 nM T59045 CL7H6I 10419448 Ki = 11000000 nM T59045 C3INT9 12896796 IC50 > 1000000 nM T59045 COG3R4 22247029 IC50 > 5000000 nM T59045 C8OP4K 10351955 Ki = 6300000 nM T59045 C6G5XN 135408704 IC50 > 1000000 nM T59045 C59TVG 44378094 Ki = 9000 nM T59045 D00YEV 5281605 IC50 = 12800000 nM T59045 D03VZF 18169 IC50 = 15500 nM T59045 D07ZBH 97472 IC50 = 15400 nM T59045 D0L7RB 16036927 IC50 = 5480 nM T67818 D01BYB 5957 EC50 = 150 nM T67818 D06ACW 6083 EC50 = 1500 nM T67818 D0S6AE 148197 EC50 > 20000 nM T67818 D0Z7FU 6133 EC50 > 2000 nM T67818 CPQ81V 171069 EC50 = 80 nM T67818 CVC6T8 440210 EC50 = 760 nM T67818 CR8K6U 1188014 IC50 = 140 nM T67818 C3LYX1 1188015 Ki >= 100000 nM T67818 CJX73P 1226686 Ki = 6000 nM T67818 C6P7VU 5311303 IC50 = 320 nM T67818 CIH51L 7283514 Ki = 400 nM T67818 CZW7U2 7283646 IC50 = 25000 nM T67818 C2I5JK 7312981 Ki = 400 nM T67818 C8RM7J 7313032 Ki = 500 nM T67818 CF8KI6 9847505 Ki = 2.5 nM T67818 CRE90Y 9955181 EC50 = 840 nM T67818 C3T8BS 10070925 IC50 = 148 nM T67818 C2F7DR 10098947 EC50 = 2630 nM T67818 CM96ZK 10168108 EC50 > 20000 nM T67818 CI9K1V 10191162 EC50 > 20000 nM T67818 CM4K6R 10303040 EC50 > 20000 nM T67818 CZE5Y1 10482694 EC50 = 80 nM T67818 C2BVH7 10601567 Ki = 17.6 nM T67818 C3L6KW 10994891 EC50 = 52 nM T67818 CJS9C0 11304851 IC50 > 25000 nM T67818 C36FVH 11409030 Ki = 91 nM T67818 C4KTZ9 11496216 Ki = 7.3 nM T67818 CO26HV 11510223 Ki = 31 nM T67818 CHB3C7 11510273 Ki = 16 nM T67818 C3AFT9 11517789 Ki = 26 nM T67818 C7ZR5X 11518174 Ki = 16 nM T67818 C2WS9Q 11531074 Ki = 28 nM T67818 CWZ3D4 11533956 Ki = 390 nM T67818 C12UVD 11541258 Ki = 260 nM T67818 C8PDH3 11549000 IC50 = 5.9 nM T67818 CT74ZJ 11560464 Ki = 7 nM T67818 CHR5C4 11562092 Ki = 4500 nM T67818 CQM17R 11562714 Ki = 300 nM T67818 C1X9UA 11575089 Ki = 172 nM T67818 C7NK4X 11575502 Ki = 36.5 nM T67818 CQIE41 11575842 Ki = 20.3 nM T67818 CMKY61 11583568 Ki = 6.6 nM T67818 CJG3K6 11604868 Ki = 7.6 nM T67818 C4G3BS 11606309 Ki = 13.3 nM T67818 CUD1J5 11611428 Ki = 8 nM T67818 CO23MC 11614523 IC50 < 1000 nM T67818 C8V0QO 11620229 Ki = 690 nM T67818 CYH54P 11626368 Ki = 29.5 nM T67818 CJVD59 11634388 IC50 = 2.2 nM T67818 CX7J8F 11636756 IC50 = 1819700.86 nM T67818 CB5OD0 11640537 Ki = 65 nM T67818 CC2R9X 11642453 Ki = 290 nM T67818 C4U5MH 11648059 Ki = 28 nM T67818 C43BEI 11656611 Ki = 4500 nM T67818 C7D4FT 11662179 Ki = 830 nM T67818 CQ6SG9 11675204 Ki = 7 nM T67818 CG3K2W 11692026 Ki = 11 nM T67818 CEU74V 11698231 Ki = 39 nM T67818 CPC34H 11699502 Ki = 13500 nM T67818 CI71BX 11699791 Ki = 18.6 nM T67818 CRPZ90 11704091 Ki = 11 nM T67818 C7QD0V 11706525 Ki = 20.7 nM T67818 CI2MT7 11706804 Ki = 200 nM T67818 C70OHZ 11711880 Ki = 8.7 nM T67818 C7OFE2 11711909 Ki = 94 nM T67818 CODM63 12000021 EC50 = 1200 nM T67818 C67WNM 13455593 EC50 = 426 nM T67818 CKB09S 16005793 IC50 = 75 nM T67818 C4E8CP 16005795 IC50 = 227 nM T67818 CR6W9O 16216480 EC50 > 20000 nM T67818 C6AQ2L 16738126 Ki = 66 nM T67818 CZ7SX0 23675739 IC50 = 3000 nM T67818 CXZ58T 24799317 EC50 = 4390 nM T67818 CKO7C2 24958669 Ki = 50 nM T67818 C7K0OA 24959029 Ki = 100 nM T67818 C0JSZ6 24959030 Ki = 120 nM T67818 CZ36UC 24959031 Ki = 130 nM T67818 CSI9Q5 24959032 Ki = 250 nM T67818 CSO73E 24959398 Ki = 250 nM T67818 C7O9KD 24959759 Ki = 140 nM T67818 CWC1K6 24959760 Ki = 290 nM T67818 CARU61 24959763 Ki = 30 nM T67818 C76JQO 24960128 Ki = 70 nM T67818 C86PJO 24960131 Ki = 20 nM T67818 C2XB7S 24960132 Ki = 60 nM T67818 C29KLZ 24960493 Ki = 60 nM T67818 CZ48MB 24960497 Ki = 30 nM T67818 CMZ9Y8 25099564 Ki = 150 nM T67818 C54AXC 25169254 Ki = 70 nM T67818 C8YV9Q 40995076 Ki = 100 nM T67818 CVC9D3 44306835 EC50 = 52 nM T67818 CTB6U8 44364208 Ki = 5.1 nM T67818 CB7T0D 44364283 Ki = 12.6 nM T67818 C0UQ9H 44364323 Ki = 35 nM T67818 C7CD3U 44425066 Ki = 540 nM T67818 C5W8JN 44425067 Ki = 650 nM T67818 CMG9D2 44425068 IC50 = 870 nM T67818 CW8BQ9 44425069 IC50 = 93.33 nM T67818 CB2C1L 44425070 Ki = 273 nM T67818 CGKL72 44425071 Ki = 706 nM T67818 C2D1MQ 44439743 EC50 > 20000 nM T67818 CW2U7Z 44439757 EC50 > 20000 nM T67818 C42YBU 44439758 EC50 > 20000 nM T67818 C0IBA3 44439765 EC50 > 20000 nM T67818 CI74KG 44448768 Ki = 5200 nM T67818 CT6N0P 44448802 Ki > 10000 nM T67818 C4U5HR 44448803 Ki = 1800 nM T67818 CP70GV 44448830 Ki > 10000 nM T67818 CO31DG 44448868 Ki > 10000 nM T67818 C4UBN8 44448870 Ki > 10000 nM T67818 CP0BD2 44448871 Ki > 10000 nM T67818 CRM3C1 44448909 Ki > 10000 nM T67818 C5Q1YK 44448911 Ki = 1200 nM T67818 CQF4Z2 44448944 Ki > 10000 nM T67818 C4HF1P 44448945 Ki > 10000 nM T67818 CVA01W 44448974 Ki = 760 nM T67818 CI96JR 44449026 Ki = 120 nM T67818 CERK23 44449075 Ki = 2700 nM T67818 CAD32B 44449077 Ki = 130 nM T67818 CQ2P9F 44449103 Ki = 200 nM T67818 C4ZEH5 44449104 Ki = 180 nM T67818 C7OX1B 44449105 Ki = 560 nM T67818 C40LXK 44449129 Ki > 10000 nM T67818 C8F3AN 44449130 Ki = 700 nM T67818 C2S8MC 44449132 Ki = 7200 nM T67818 C6IV9P 44449164 Ki > 10000 nM T67818 CTF47A 44449165 Ki = 270 nM T67818 CTKW57 44449166 Ki > 10000 nM T67818 C5YI3T 44449191 Ki > 10000 nM T67818 C9YID2 44449195 Ki = 960 nM T67818 CMHK57 44562602 IC50 > 25000 nM T67818 C4VGQ9 44562603 IC50 > 25000 nM T67818 CLJX37 44562653 Ki = 300 nM T67818 CS3DV0 44562758 Ki = 300 nM T67818 COV1S4 44562759 Ki = 500 nM T67818 CRU78M 44562760 IC50 = 6000 nM T67818 CQSC98 44562761 Ki = 100 nM T67818 C3FS9P 44562795 Ki = 400 nM T67818 C2M8EJ 44562796 Ki = 200 nM T67818 C1YGU0 44562797 Ki = 800 nM T67818 C7QN9K 44562836 IC50 > 25000 nM T67818 CUC87A 44562837 IC50 = 10000 nM T67818 CRD29T 44562838 IC50 > 25000 nM T67818 C4M6UO 44562839 IC50 > 25000 nM T67818 C8IKO9 44563234 IC50 > 25000 nM T67818 CV69BH 44563235 Ki = 100 nM T67818 CZD86A 46228890 EC50 = 420 nM T67818 C4U6LZ 46228892 EC50 = 460 nM T67818 CWR97Z 46228944 EC50 = 11 nM T67818 CI83JW 46229259 EC50 = 1.89 nM T67818 CQNZ48 46241018 IC50 = 4900 nM T67818 CVP5D0 46241232 IC50 = 29000 nM T67818 CPZ83K 46911434 IC50 = 1600 nM T67818 CF4DN0 46911436 IC50 = 300 nM T67818 CL2U0Q 46911481 Ki = 600 nM T67818 CU0XK3 49797754 Ki = 640 nM T67818 C0IC7Y 49797755 Ki = 760 nM T67818 C6K2YC 49797777 IC50 = 15800 nM T67818 C1D8NS 49797778 IC50 = 5000 nM T67818 CTQ4H0 49798096 IC50 > 25000 nM T67818 C0ICW7 49798097 Ki = 2500 nM T67818 CNZ54V 49798145 Ki = 400 nM T67818 C36ALC 49798146 IC50 > 25000 nM T67818 CPV84E 49798147 IC50 > 25000 nM T67818 C30CIT 49856886 EC50 = 300 nM T67818 C2O6TI 49856888 EC50 >= 30000 nM T67818 CJGE25 49857082 EC50 = 30000 nM T67818 CKI5H9 51032193 IC50 = 10200 nM T67818 CR98BF 53350233 IC50 = 2.5 nM T67818 CP87YH 53350234 Ki = 12 nM T67818 CJ2RM6 56673378 EC50 = 9000 nM T67818 C1I4YV 59128840 Ki = 70 nM T67818 CYQ3S9 59128841 Ki = 21 nM T67818 CKP5V0 59128886 Ki = 207 nM T67818 C1U8JL 59128890 Ki = 11 nM T67818 CI5P7T 59128900 Ki = 12 nM T67818 CRS58Y 59128945 Ki = 435 nM T67818 CL2VD6 59128964 Ki = 45 nM T67818 C3SYF6 59128997 Ki = 31 nM T67818 CY3JA1 59129000 Ki = 1500 nM T67818 CSHK27 59129016 Ki = 410 nM T67818 CPC0R9 59129017 Ki = 2900 nM T67818 CI8U6F 59129057 Ki = 7 nM T67818 CI3LA5 59129071 Ki = 25 nM T67818 CK36PG 59129092 Ki = 59 nM T67818 C94KLF 59129106 Ki > 36000 nM T67818 CX5J7S 59129109 Ki = 186 nM T67818 CUIW36 59129118 Ki = 6 nM T67818 CC86AI 59275020 Ki = 15 nM T67818 C8Z5FQ 60150614 IC50 = 0.12 nM T67818 CM4Y7B 66554126 Ki = 27000 nM T67818 C81MOI 66554204 Ki = 42000 nM T67818 CS6WU1 66554206 Ki >= 100000 nM T67818 C28ZIU 66554207 Ki = 45000 nM T67818 CG8ET1 66554279 IC50 = 130 nM T67818 CR7W0Y 66855824 Ki > 20000 nM T67818 CG7DL9 68527699 Ki = 98 nM T67818 C4QOM2 68528196 Ki = 68 nM T67818 CME65J 68528291 Ki = 69 nM T67818 CUFB01 68528415 Ki = 322 nM T67818 C5QB6P 68528423 Ki = 150 nM T67818 C4B8KQ 68529738 Ki = 30 nM T67818 CF59TE 68529945 Ki = 75 nM T67818 CAXP47 68530003 Ki = 55 nM T67818 CH49EF 68530011 Ki = 190 nM T67818 C9UQ0F 68530013 Ki = 54 nM T67818 C4VFI2 68530100 Ki = 20 nM T67818 CB1US3 68530232 Ki = 60 nM T67818 CD2H8Q 68530233 Ki = 145 nM T67818 CS4NA7 68530266 Ki = 21 nM T67818 CV87OT 68530361 Ki = 77 nM T67818 C2S6UR 68530403 Ki = 34 nM T67818 CTS25B 68531201 Ki = 84 nM T67818 CG6Y9J 68531462 Ki = 7 nM T67818 C9UL7Q 68531481 Ki = 25 nM T67818 CXY86G 68531609 Ki = 121 nM T67818 CF4UT2 68531763 Ki = 87 nM T67818 CXH92L 68531887 Ki = 37 nM T67818 C2MK3E 68531895 Ki = 18 nM T67818 CLT8G2 68531914 Ki = 7 nM T67818 C23XLR 68531926 Ki = 137 nM T67818 C9ASJ6 68532402 Ki = 169 nM T67818 C2QHI1 68533081 Ki = 3000 nM T67818 C7F1NS 68533208 Ki = 175 nM T67818 CG1KM6 68533209 Ki = 176 nM T67818 C97HDS 68533305 Ki = 11 nM T67818 C85NIY 68533570 Ki = 16 nM T67818 CD12UA 68533659 Ki = 33 nM T67818 C7DYW9 68533683 Ki = 18 nM T67818 CZP0V6 68533690 Ki = 41 nM T67818 CL4JB2 68533783 Ki = 48 nM T67818 CKY5R1 68533937 Ki = 47 nM T67818 C1I6RU 68534835 Ki = 15 nM T67818 CDR8N4 68534837 Ki = 29 nM T67818 CD0NT4 68534854 Ki = 52 nM T67818 CL0C8B 68534894 Ki = 128 nM T67818 C09ONY 68534915 Ki = 11 nM T67818 CMB36I 70683606 EC50 = 800 nM T67818 C78RVE 70691003 Ki = 10000 nM T67818 C5Y4ST 70694092 EC50 = 800 nM T67818 CSK4A9 71449106 Ki = 330 nM T67818 CZS8T5 71449107 Ki = 3.6 nM T67818 CJK95G 71450314 EC50 = 13000 nM T67818 CJ8ZM1 71450315 EC50 = 300 nM T67818 CF9O0M 71452656 Ki = 430 nM T67818 CQ24IJ 71452712 IC50 = 367 nM T67818 CT93PB 71458038 Ki = 80 nM T67818 C1A6TZ 71461640 Ki = 45 nM T67818 C6VWM7 71574468 Ki > 5000 nM T67818 CK6NC9 71574469 Ki = 171 nM T67818 CXLT45 71574470 Ki > 5000 nM T67818 CB0IR9 71574471 Ki = 607 nM T67818 C6SR9Y 71574567 Ki = 313 nM T67818 C0RDU7 71574659 Ki = 506 nM T67818 C6V3YB 71574660 Ki = 571 nM T67818 CU4ZF1 71574661 Ki = 644 nM T67818 CPUM34 71574662 Ki > 5000 nM T67818 C76RHK 71574753 Ki > 5000 nM T67818 C5FH4K 71574756 Ki = 2000 nM T67818 CI8KH6 71574846 Ki > 5000 nM T67818 C8D7PM 71574847 Ki > 5000 nM T67818 CU9ZS7 71625565 Ki = 1396 nM T67818 CP09ZW 71625681 Ki = 8041 nM T67818 C0XHQ2 71625682 Ki = 592 nM T67818 CRD4I9 71625797 Ki = 17 nM T67818 CD53PN 71625914 Ki = 163 nM T67818 C21XNQ 71625915 Ki = 989 nM T67818 C0SJ8P 71655365 Ki = 2500 nM T67818 CU7B3E 71655366 Ki = 19 nM T67818 C7VZI0 71655367 Ki = 23 nM T67818 CQNZ32 71655430 Ki = 870 nM T67818 CCX9J6 71655431 Ki = 2730 nM T67818 CNES03 71655432 Ki = 10 nM T67818 C8DF7S 71655434 Ki = 27 nM T67818 CM05LO 71655491 Ki = 55 nM T67818 CZQ7U0 71655492 Ki = 250 nM T67818 C4E9OK 71655493 Ki = 670 nM T67818 C5CSZ0 71655494 Ki = 18 nM T67818 C8Z9UV 71655495 Ki = 21 nM T67818 CS7KG1 71655496 Ki = 340 nM T67818 CH9MO6 71655560 Ki = 275 nM T67818 C3A2BL 71655561 Ki = 90 nM T67818 CY2I5K 71719720 EC50 = 2.6 nM T67818 CJM56I 72725470 Ki = 620 nM T67818 CU2SK3 72725471 Ki = 1700 nM T67818 CV96IX 72725472 Ki = 560 nM T67818 CKM9X1 72725521 Ki = 1100 nM T67818 CO4XM2 72725522 Ki = 1200 nM T67818 CLEK07 72725575 Ki = 1040 nM T67818 CK9S6U 72725576 Ki = 2200 nM T67818 CB6E5C 72725577 Ki = 3400 nM T67818 CP1A7R 72725639 Ki = 3700 nM T67818 CCUG93 72736558 IC50 = 10.7 nM T67818 CSD89Y 72736559 Ki = 28.7 nM T67818 C0OTN6 72736560 IC50 = 346 nM T67818 C1HO5L 72736732 Ki = 253 nM T67818 CIV10M 72736733 Ki = 4.6 nM T67818 C64CYB 72736734 Ki = 12.8 nM T67818 CXY03I 72736735 Ki = 5.8 nM T67818 C7TFZ4 72737647 IC50 = 0.08 nM T67818 CL4J1B 72737648 IC50 = 0.02 nM T67818 C8IGS1 72737649 IC50 = 0.14 nM T67818 C7HCY0 73050925 IC50 = 0.2 nM T67818 CW9TV6 73051080 IC50 = 9.8 nM T67818 C1H7JU 73051081 IC50 = 3.6 nM T67818 CV64UL 73051082 IC50 = 1.6 nM T67818 C8G1PR 73051234 IC50 = 0.34 nM T67818 C2GNQ1 73051382 IC50 = 0.32 nM T67818 C64DKY 73051538 Ki = 66 nM T67818 CCG4F3 73051864 IC50 = 0.63 nM T67818 CERM21 73052662 IC50 = 0.23 nM T67818 CO7G4L 73052824 IC50 = 0.37 nM T67818 C2FW9M 73052977 IC50 = 0.19 nM T67818 C1HY0Q 73052978 IC50 = 0.04 nM T67818 C58VAC 73053120 IC50 = 0.21 nM T67818 CW28PS 73053272 IC50 = 1.5 nM T67818 CJF1P4 73345772 EC50 = 590 nM T67818 C02HLS 73345961 Ki = 7 nM T67818 C3DV7K 73347252 EC50 = 1890 nM T67818 C9QR2A 73347373 EC50 = 74 nM T67818 CL0X8W 73347374 EC50 = 150 nM T67818 C8HTZ1 73347375 EC50 = 3000 nM T67818 C8H0CE 73348762 EC50 = 7 nM T67818 C1I6HS 73348763 EC50 = 33 nM T67818 C7C4UW 73348769 EC50 = 23 nM T67818 C3KN0U 73348774 EC50 = 0.4 nM T67818 C52QYE 73350589 Ki = 8 nM T67818 CQ84GJ 73350590 Ki = 8 nM T67818 C6HS9D 73350591 Ki = 195 nM T67818 CB8VW7 73351851 EC50 = 158 nM T67818 CLXM46 73351984 EC50 = 600 nM T67818 CJO1P5 73351985 EC50 = 200 nM T67818 C2K1LV 73352098 Ki = 5 nM T67818 CEO3T7 73352099 Ki = 8 nM T67818 C2D7HR 73352100 Ki = 13 nM T67818 C9CWV3 73353445 EC50 = 950 nM T67818 CU98ZX 73353558 Ki = 4850 nM T67818 C5FU8W 73353559 Ki = 12 nM T67818 CX13RQ 73354954 EC50 = 2500 nM T67818 COQJ62 73356385 EC50 = 9 nM T67818 C5PI9L 73356611 Ki = 11 nM T67818 CJOU70 73671602 Ki = 57 nM T67818 CZ9UW5 90034698 IC50 = 0.23 nM T67818 CR4FU2 90035491 IC50 = 3100 nM T67818 CC2W9Y 90062960 IC50 = 0.51 nM T67818 C7F0MJ 90062981 IC50 = 0.37 nM T67818 C6T2YH 90062983 IC50 = 0.57 nM T67818 CAMF46 90062985 IC50 = 0.15 nM T67818 C9CIZ7 90062986 IC50 = 0.13 nM T67818 CT1V0N 90062993 IC50 = 300 nM T67818 CGCH61 90062998 IC50 = 1.06 nM T67818 C62VIS 90062999 IC50 = 390 nM T67818 C09WGQ 90063071 IC50 = 0.05 nM T67818 C7G6PA 90063075 IC50 = 1.96 nM T67818 CI56XS 90063103 IC50 = 0.52 nM T67818 CMAQ85 90070531 Ki = 6 nM T67818 CE7ZY9 90078528 IC50 = 0.15 nM T67818 CES8C1 90078535 IC50 = 180 nM T67818 C2NS8T 90078572 IC50 = 0.13 nM T67818 C3OP4V 90643794 IC50 > 150 nM T67818 C7G5ZR 90643795 IC50 > 150 nM T67818 CI40GL 90643796 IC50 = 0.17 nM T67818 C0TAD6 90643797 IC50 = 0.06 nM T67818 CHI5B2 90643798 IC50 = 0.03 nM T67818 C10UYN 90643799 IC50 = 0.08 nM T67818 C7IBN8 90643800 IC50 = 0.04 nM T67818 CW5P2G 90643801 IC50 = 4.6 nM T67818 CV79FU 90656740 Ki = 6.2 nM T67818 CZK9N0 90656741 Ki = 20 nM T67818 C8MI1O 90656742 IC50 = 2.3 nM T67818 CCX80K 90656743 Ki = 343 nM T67818 C6AW1H 90656744 Ki = 511 nM T67818 C03ZVE 90656745 Ki = 49 nM T67818 C4WO7N 90656746 IC50 = 2.7 nM T67818 C85TRU 118130556 IC50 = 0.16 nM T67818 CK9R4M 118130678 IC50 = 140 nM T67818 C0NZW4 118365897 IC50 = 2.3 nM T67818 C3LW4B 118365898 IC50 = 1.8 nM T67818 CL8NJ6 118365906 IC50 = 0.39 nM T67818 C37ALN 118365922 IC50 = 0.04 nM T67818 CNV9E6 118365942 IC50 = 230 nM T67818 CL1AO4 118365947 IC50 = 0.03 nM T67818 CPZ45X 118365960 IC50 = 0.13 nM T67818 C0SYW2 118365962 IC50 = 0.33 nM T67818 CM1IN7 118365990 IC50 = 0.37 nM T67818 CI3UJ8 118365999 IC50 = 0.08 nM T67818 CU0N5V 118707544 IC50 = 0.14 nM T67818 C78INB 118725181 EC50 = 7 nM T67818 CM8N4I 122195891 EC50 = 2.6 nM T67818 CULF46 122195892 EC50 = 30 nM T67818 CC2JO4 122195893 EC50 = 730 nM T67818 C9HK0N 122195894 EC50 = 37 nM T67818 CZ1XL2 122195895 EC50 = 90 nM T67818 CKR2L7 127038948 IC50 = 360 nM T67818 CBXP14 127038950 IC50 = 1020 nM T67818 CN7C8A 127039315 IC50 = 2150 nM T67818 C2N9XI 127039918 IC50 = 5200 nM T67818 CF0M8H 127039999 IC50 = 160 nM T67818 CV8XS2 127040346 IC50 = 9600 nM T67818 CIMH26 127040665 IC50 = 6300 nM T67818 C7RQT4 127040675 IC50 = 4210 nM T67818 CNPL48 127040996 IC50 = 7370 nM T67818 CH42ZI 127040998 IC50 = 2240 nM T67818 CV4AL5 127041004 IC50 = 2650 nM T67818 C9ON2A 127041006 IC50 = 1970 nM T67818 CKB30T 127041008 IC50 = 8800 nM T67818 CHIG78 132574706 IC50 = 4550 nM T67818 CJXA12 134611894 Ki < 1000 nM T67818 C3WMJ7 136074319 IC50 = 0.57 nM T67818 CMP2F1 136074320 IC50 = 160 nM T67818 CTXB02 136074321 IC50 = 0.3 nM T67818 C1VRT2 136074322 IC50 = 260 nM T67818 C6ZB1D 137632198 IC50 = 7650 nM T67818 C4GA0J 137641946 IC50 = 25000 nM T67818 C7O3US 137643396 IC50 = 5480 nM T67818 CUR8V1 137648798 IC50 = 2720 nM T67818 CGA95F 145980072 IC50 = 2410 nM T67818 CGL5O4 145981034 IC50 = 820 nM T67818 CXP6G9 145982090 IC50 = 12920 nM T67818 CC7IW1 145982935 IC50 = 210 nM T67818 CJ10ZX 145984169 IC50 = 7050 nM T67818 C0GD5Q 145989182 IC50 = 7190 nM T67818 C1V4TN 145990707 IC50 = 9980 nM T67818 C0G6ST 145991143 IC50 = 620 nM T67818 CY28NJ 145991243 IC50 = 12520 nM T67818 CF4CT9 145993655 IC50 = 7530 nM T67818 D01APA 66855377 Ki > 20000 nM T67818 D02HAL 6031 EC50 > 100000 nM T67818 D03ERS 44448831 Ki = 0.78 nM T67818 D05MXI 42611190 IC50 > 10000 nM T67818 D05NWF 6022 EC50 = 14 nM T67818 D07MTB 11510579 Ki = 6 nM T67818 D07QYU 4881 EC50 = 1000 nM T67818 D08DXA 23675622 IC50 = 17600 nM T67818 D09DLY 989142 Ki = 4900 nM T67818 D0BB0O 121990 EC50 = 1.27 nM T67818 D0D5NP 10894633 Ki = 76 nM T67818 D0E9DE 71655433 Ki = 7 nM T67818 D0G8KA 24958668 Ki = 90 nM T67818 D0KF2P 44126037 Ki > 20000 nM T67818 D0NJ7Y 46911435 Ki = 140 nM T67818 D0U1OJ 5310983 EC50 = 34 nM T67818 D0U8HD 162565 EC50 = 770 nM T67818 D0V4GQ 5310996 EC50 = 1270 nM T67818 D0W8WZ 24743975 Ki = 10 nM T47768 D00KHM 16362 IC50 = 372 nM T47768 D00UYE 4058 IC50 = 315 nM T47768 D01KQA 5311304 Ki = 0.89 nM T47768 D02NSF 5284604 Ki = 1.79 nM T47768 D02RXG 6918287 EC50 = 1.7 nM T47768 D03DIG 5284371 IC50 = 105 nM T47768 D03SKD 5284603 Ki = 12 nM T47768 D03YVO 5361917 Ki = 5.48 nM T47768 D04JEE 4946 EC50 > 5011.87 nM T47768 D04JHN 5284570 Ki = 0.28 nM T47768 D04QWE 5359371 Ki = 0.48 nM T47768 D05DVP 5717 IC50 > 10000 nM T47768 D05GKD 33741 EC50 = 1000 nM T47768 D05VIL 5284594 Ki = 0.24 nM T47768 D09OJQ 4095 IC50 = 4.1 nM T47768 D09ZXR 11250029 EC50 = 1 nM T47768 D0CQ0Z 33630 Ki = 867 nM T47768 D0CS2F 3955 Ki = 0.53 nM T47768 D0D1AL 3559 EC50 > 10000 nM T47768 D0D7KC 5488548 Ki = 0.3162 nM T47768 D0D8DD 41693 EC50 = 1.3 nM T47768 D0E1WI 3345 EC50 = 0.51 nM T47768 D0I0DL 3689 IC50 > 1000 nM T47768 D0P6VV 3033053 EC50 = 38 nM T47768 D0PG8O 5360515 Ki = 0.07 nM T47768 D0T3HY 5359272 IC50 = 0.13 nM T47768 D0WE3O 5288826 Ki = 0.14 nM T47768 D0X3FX 5284596 Ki = 0.23 nM T47768 D0X5KF 5284569 Ki = 9.5 nM T47768 D0X9RG 5361092 Ki = 0.12 nM T47768 D00HBR 5486554 Ki = 0.19 nM T47768 D01UXW 5360621 Ki = 12.9 nM T47768 D03PJU 62156 EC50 = 0.0049 nM T47768 D03TBJ 11848225 Ki = 0.7 nM T47768 D06ENM 66553195 Ki = 6 nM T47768 D06EXA 128563 Ki > 1000 nM T47768 D07TQN 179340 EC50 = 60000 nM T47768 D07YHM 44129648 Ki = 16.4 nM T47768 D09ALE 60768 Ki = 22 nM T47768 D0K5HI 5311424 Ki = 1860 nM T47768 D0LI1C 44469321 IC50 > 10000 nM T47768 D0N1HW 5311200 Ki > 10000 nM T47768 D0Q3PD 54732242 Ki = 1.1 nM T47768 D0R0EF 24772484 IC50 = 460 nM T47768 D0T0ZW 11667832 Ki = 0.052 nM T47768 D0V5WL 443363 IC50 = 13 nM T47768 D0W4YO 16131448 Ki = 270 nM T47768 D0C2QF 9906198 Ki = 0.043 nM T47768 D0M1YN 5311194 Ki > 400 nM T47768 D0N1RG 9805452 Ki = 51 nM T47768 D00ACC 9844019 Ki > 400 nM T47768 D04XCQ 10099811 Ki = 4000 nM T47768 D06DZI 107780 Ki > 10000 nM T47768 D0K5KL 119029 IC50 = 2.1 nM T47768 D0LX5D 5487663 EC50 = 1 nM T47768 D0M7BW 3505 Ki = 0.36 nM T47768 CAG0J1 5523 EC50 = 1300 nM T47768 C5XI4O 5603 IC50 = 14 nM T47768 C06VCS 5750 Ki = 920 nM T47768 C5H9CN 9287 Ki > 10000 nM T47768 CZC17M 9669 Ki = 3.9 nM T47768 C1F3WP 32414 IC50 = 1100 nM T47768 C6E8DS 62513 Ki > 10000 nM T47768 CBGO28 70419 Ki = 500 nM T47768 CX5R6B 71420 IC50 = 1.5 nM T47768 CYKE31 104920 IC50 = 3530 nM T47768 C3CU5L 107772 EC50 = 3.981 nM T47768 C9NJK8 114876 Ki = 594 nM T47768 CQYC47 121999 Ki = 40.6 nM T47768 CDM08R 124716 Ki = 0.089 nM T47768 C7USG2 132913 Ki = 80 nM T47768 CB8Y9H 134131 IC50 = 1.1 nM T47768 C4LEU1 191408 Ki = 5900 nM T47768 C3HB4V 416359 EC50 = 2183 nM T47768 C27OGF 449698 Ki = 0.07 nM T47768 CBLC72 457967 EC50 = 16000 nM T47768 C5HTX2 607612 EC50 = 2280 nM T47768 C97LRS 620160 EC50 = 4720 nM T47768 CR45EB 644177 Ki > 1000 nM T47768 C3VFW0 715222 EC50 = 150 nM T47768 CPW2B6 715224 EC50 = 1120 nM T47768 CZN6S9 743974 EC50 > 100000 nM T47768 CLZ04O 746650 EC50 = 4000 nM T47768 CY4FS5 746662 EC50 > 30000 nM T47768 C6BDH3 780684 EC50 = 39000 nM T47768 CB27WS 849733 IC50 > 10000 nM T47768 C0QU4L 972358 EC50 = 19000 nM T47768 C8H0KW 1009511 EC50 = 2000 nM T47768 C4U2MZ 1044308 EC50 = 5000 nM T47768 C6B0TP 1121183 EC50 = 6100 nM T47768 C7ZB8J 1144657 EC50 > 30000 nM T47768 CB6L7E 1878753 EC50 > 100000 nM T47768 CX8KH4 2297178 EC50 = 3000 nM T47768 C7DFA2 2724431 EC50 = 17 nM T47768 CP69WS 2750525 EC50 = 750 nM T47768 CAO06Q 2796048 IC50 = 4590 nM T47768 CLSF10 2823239 IC50 = 17000 nM T47768 CGET70 2832042 EC50 = 6380 nM T47768 C1MCQ6 2912831 EC50 > 100000 nM T47768 C2UGQ1 2913055 EC50 = 9910 nM T47768 CLXC53 3000341 Ki = 118 nM T47768 CAQ2J0 3034396 Ki = 161 nM T47768 C2TAD3 3036289 Ki = 290 nM T47768 CLB7W5 3037886 Ki = 3.8 nM T47768 CH0Z2R 3037926 Ki = 0.16 nM T47768 C5HDK8 3041260 Ki = 0.02 nM T47768 C5K7GJ 3054741 EC50 = 21 nM T47768 C8OHF0 3081578 Ki = 23.8 nM T47768 CMKU43 3086068 Ki = 38 nM T47768 CZHC01 3112394 EC50 > 30000 nM T47768 CDIN98 3132840 EC50 = 1100 nM T47768 CJ6D8N 3342390 Ki = 306 nM T47768 CQ6MW0 3655995 Ki = 91.1 nM T47768 C0YXV3 3676358 Ki > 10000 nM T47768 CC3DM1 3955796 EC50 > 10000 nM T47768 CT52BI 4247619 EC50 = 10000 nM T47768 CXO48E 4353400 EC50 = 4000 nM T47768 CY7LK9 4491166 Ki = 0.78 nM T47768 CANE93 4545429 Ki = 53 nM T47768 CK07BP 5030548 EC50 = 1120 nM T47768 CJS15P 5091282 EC50 = 2890 nM T47768 C14LHW 5172692 EC50 = 6000 nM T47768 C2O3TW 5282407 IC50 = 2410 nM T47768 CJX28Y 5311003 Ki = 7.3 nM T47768 CLW4B1 5311340 Ki = 102 nM T47768 C6HY1P 5361918 Ki = 7.943 nM T47768 CY7P2R 5408233 EC50 = 32500 nM T47768 C2HPQ4 5462505 Ki = 1.1 nM T47768 C17RBP 5486940 Ki = 0.01 nM T47768 CJ7IE6 5487695 Ki = 85.6 nM T47768 CCMZ86 5491688 Ki = 1.4 nM T47768 CZ4TM3 5492619 Ki = 1910 nM T47768 CI7L4R 5492830 Ki = 305 nM T47768 C9LJ2K 5493351 Ki = 0.769 nM T47768 CJQN51 6438353 Ki = 1.9 nM T47768 C5AL8S 6445230 EC50 = 0.72 nM T47768 CQML02 6603856 Ki = 34.7 nM T47768 CM6VF8 6734379 IC50 = 2285 nM T47768 CFTO93 6918704 Ki = 0.18 nM T47768 CD49UV 9797246 Ki = 233 nM T47768 CNO0W4 9799433 Ki = 1.07 nM T47768 C8ANR0 9801260 IC50 = 632 nM T47768 C5RNW7 9801830 IC50 = 2064 nM T47768 C3V7JB 9802297 Ki > 4652 nM T47768 CPG57N 9803475 Ki > 400 nM T47768 C5Z2KM 9805944 Ki = 0.6 nM T47768 CPRQ41 9806459 Ki >= 2000 nM T47768 CX7DO4 9806799 Ki = 1069 nM T47768 C1TQM8 9809562 Ki = 0.143 nM T47768 CVL4W8 9820950 Ki = 855 nM T47768 CJ72XV 9822639 Ki = 35 nM T47768 CXV1R9 9822756 IC50 = 1240 nM T47768 CE6NF9 9823363 IC50 > 10000 nM T47768 C70KEP 9824565 Ki = 249 nM T47768 CR54GJ 9824976 Ki > 890 nM T47768 CP38OJ 9825316 Ki = 172 nM T47768 C07FWV 9830361 Ki = 1320 nM T47768 CDT81N 9838022 Ki = 160 nM T47768 CYN53X 9838412 Ki = 286 nM T47768 CW1T4D 9839245 Ki = 0.31 nM T47768 CX40CL 9840199 Ki = 0.1 nM T47768 C4QFZ6 9841259 IC50 = 3800 nM T47768 CKVQ31 9843334 Ki = 2763 nM T47768 C6Y7NA 9844540 Ki = 256 nM T47768 CJ8LT7 9848518 IC50 > 10000 nM T47768 CH06GL 9848989 IC50 = 1.7 nM T47768 CKD2H4 9848990 Ki = 0.09 nM T47768 CME87B 9849361 Ki = 0.031 nM T47768 CHM93P 9862850 EC50 = 551 nM T47768 CBMN05 9865332 Ki = 52 nM T47768 CLQ6Z8 9866158 Ki = 37 nM T47768 CL26PE 9866175 Ki > 890 nM T47768 CT2C6K 9870702 IC50 > 10000 nM T47768 CQ4LC2 9872676 Ki = 1400 nM T47768 C3LOJ7 9872857 Ki = 195 nM T47768 CEO0M2 9880173 Ki = 426 nM T47768 CLSP49 9881709 IC50 = 56 nM T47768 CPYK08 9887195 IC50 = 3300 nM T47768 C67GMC 9888235 Ki = 3650 nM T47768 CB8G9J 9889993 Ki = 0.26 nM T47768 CJF8C2 9890982 EC50 = 18.8 nM T47768 C1VM4H 9902583 Ki = 716 nM T47768 C5BC4P 9902874 Ki = 959 nM T47768 CUN81Q 9905249 Ki > 10000 nM T47768 CX3CM8 9905428 Ki = 29.9 nM T47768 C4X6PY 9909946 EC50 = 2 nM T47768 CB6C8L 9911987 Ki = 88 nM T47768 C2TE5X 9922658 Ki = 3 nM T47768 C4NJ0W 9923726 Ki = 1402 nM T47768 CIUE54 9924406 Ki = 6.4 nM T47768 C5HN0J 9925137 Ki = 9.5 nM T47768 C7L4MX 9927776 EC50 = 591 nM T47768 CZT2J0 9927928 Ki = 46.97 nM T47768 C26DMO 9928857 Ki = 25.8 nM T47768 CM3B5E 9932532 Ki > 890 nM T47768 C2U8XH 9932834 Ki = 22 nM T47768 CYZW21 9932852 EC50 = 2445 nM T47768 C9MK3B 9934232 Ki = 595 nM T47768 CUBQ95 9937777 Ki = 436 nM T47768 CO7BI9 9940052 Ki = 36.9 nM T47768 C4FD7V 9947044 Ki = 12.8 nM T47768 C5S3RH 9949205 Ki = 1.72 nM T47768 CUE9Z8 9951118 Ki = 0.3162 nM T47768 CKNZ54 9951665 Ki = 5040 nM T47768 COFT18 9951673 Ki = 609 nM T47768 C3GXH0 9954388 Ki = 7.2 nM T47768 CPZ4B5 9956370 Ki = 226 nM T47768 CT8C2X 9958643 Ki = 616 nM T47768 CW02IS 9959144 Ki = 0.16 nM T47768 C1B2JR 9976188 Ki = 47.7 nM T47768 C2GI1Q 9984781 Ki = 219.16 nM T47768 CD0IS5 9985476 Ki > 30000 nM T47768 C2WJL0 9990996 Ki = 21 nM T47768 CAGL19 9997843 Ki = 3.4 nM T47768 CN2F1U 10001960 IC50 = 1510 nM T47768 CQL12P 10004545 Ki > 2000 nM T47768 CL9QS0 10004950 IC50 = 0.9 nM T47768 C9CP0Q 10005080 Ki = 47 nM T47768 CQ43EZ 10016044 Ki = 0.16 nM T47768 CV7R9F 10020040 Ki > 10000 nM T47768 C4N8YE 10020165 Ki = 14.4 nM T47768 CL38DM 10021831 Ki = 0.013 nM T47768 C25DYT 10022859 Ki = 5.9 nM T47768 C0O9EM 10024658 IC50 = 2716 nM T47768 C1PGE2 10031234 Ki = 130 nM T47768 CFOK60 10042904 Ki = 8 nM T47768 CC60VS 10052051 Ki = 0.16 nM T47768 C4CXP1 10053267 Ki = 6.5 nM T47768 C8WE1N 10055958 IC50 = 225 nM T47768 CS3UK5 10074239 Ki = 43.8 nM T47768 CO8P3K 10076169 Ki = 9 nM T47768 CM34WV 10077545 Ki > 4500 nM T47768 CQVA98 10078468 Ki = 0.16 nM T47768 CZ5H9X 10093250 Ki = 322 nM T47768 CV1OU6 10109140 Ki = 1.9 nM T47768 C7YCF1 10109899 Ki = 28 nM T47768 CJNE19 10110916 Ki = 5545 nM T47768 C0PC9A 10113006 Ki = 39.6 nM T47768 CL5MY1 10116470 Ki = 276 nM T47768 CB4P7L 10116719 Ki = 163 nM T47768 C40BMF 10133108 Ki = 208 nM T47768 C2WZ9G 10133332 Ki = 1237 nM T47768 CP1SO7 10134077 Ki = 448 nM T47768 CEG0M4 10134217 Ki = 748 nM T47768 C3ZTU0 10137134 Ki = 2454 nM T47768 C83KDV 10137876 Ki = 86 nM T47768 C8E9KP 10139672 Ki = 182 nM T47768 CVRZ09 10141332 Ki = 237 nM T47768 CT1B5J 10142188 Ki = 22.4 nM T47768 CKCW48 10143870 Ki = 0.44 nM T47768 CI3PJ6 10149623 Ki > 10000 nM T47768 CQGE97 10150001 Ki = 488 nM T47768 CF85VW 10150089 Ki > 10000 nM T47768 C76SOW 10150260 Ki = 1654 nM T47768 CRC46J 10154739 Ki = 435 nM T47768 CKN3A8 10154848 Ki = 395 nM T47768 CFIL01 10155966 Ki = 94 nM T47768 CIO6U3 10156336 Ki = 2165 nM T47768 CP53IB 10156591 Ki = 9 nM T47768 CI1U4Z 10156821 Ki = 514 nM T47768 CTO0N5 10158555 Ki = 692 nM T47768 CG51TX 10159203 Ki = 65 nM T47768 CWM2X6 10160920 Ki = 38 nM T47768 C8ZA6U 10164835 Ki = 337 nM T47768 C67SZC 10171702 Ki > 10000 nM T47768 CB57JZ 10171862 Ki = 12 nM T47768 CDV15J 10172398 Ki = 152 nM T47768 CJN21A 10178311 Ki = 279 nM T47768 CHN4G6 10178563 Ki = 199 nM T47768 CK5HG3 10179322 Ki > 465 nM T47768 CHC6K9 10179323 Ki > 465 nM T47768 C2SP7U 10183838 Ki = 980 nM T47768 CUE8P2 10184592 Ki = 451 nM T47768 C2PTU7 10185016 Ki = 9643 nM T47768 C2QF7B 10185709 Ki = 644 nM T47768 CNZL85 10193971 Ki = 5551 nM T47768 CN79QX 10194236 Ki = 1967 nM T47768 CWC8L1 10199945 IC50 = 3500 nM T47768 C85DFV 10201299 Ki > 465 nM T47768 CH40KY 10202108 Ki = 27 nM T47768 CZ4N2S 10205966 Ki = 608 nM T47768 C9ZCT0 10206319 Ki = 282 nM T47768 C1HP9A 10206324 Ki = 1281 nM T47768 C31PWM 10206991 Ki = 393 nM T47768 C1J2WS 10207509 Ki = 53 nM T47768 C02IUS 10214859 Ki = 850 nM T47768 CYB0H9 10221539 IC50 = 3100 nM T47768 CZ5S1P 10224082 Ki = 50118.72 nM T47768 CRGJ86 10224456 IC50 > 10000 nM T47768 CM27FK 10225083 Ki = 34 nM T47768 C0I9TS 10226635 Ki = 1.01 nM T47768 C2XQR3 10227005 Ki = 2.99 nM T47768 C2MQS5 10227615 Ki > 4652 nM T47768 CJW0B6 10228465 Ki = 630 nM T47768 CTF5Z8 10229655 Ki = 0.24 nM T47768 CZ0C5T 10252647 Ki = 4042 nM T47768 CR4C1F 10253032 Ki = 304 nM T47768 CLKQ39 10255149 EC50 = 161 nM T47768 C4RX1A 10256503 Ki = 15 nM T47768 CH31DX 10267394 Ki > 10000 nM T47768 C58WLB 10273422 Ki = 289 nM T47768 C6YKB9 10273543 Ki > 1000 nM T47768 C8PL7B 10274330 Ki = 25 nM T47768 CR1HX2 10275388 Ki = 267 nM T47768 CSO8D7 10276738 Ki = 21 nM T47768 CO2M7L 10278214 Ki = 104 nM T47768 CUF17K 10279008 Ki = 103 nM T47768 C89KBW 10286378 Ki > 10000 nM T47768 CDP01X 10286440 Ki = 8067 nM T47768 C1FE9H 10286996 Ki = 4245 nM T47768 CJ14VU 10291377 Ki = 1071 nM T47768 C61OKS 10292091 Ki = 909 nM T47768 CKO2I1 10297473 Ki > 465 nM T47768 CTG5B1 10300866 Ki = 717 nM T47768 CV0T3H 10301207 Ki = 27 nM T47768 CF4VO2 10308746 Ki = 4000 nM T47768 CU89JD 10314060 Ki > 10000 nM T47768 CFHC64 10315026 Ki = 1.63 nM T47768 CQD21X 10315939 Ki = 5.26 nM T47768 C1ENR2 10323169 Ki = 37 nM T47768 CA4KJ5 10323346 Ki = 29.3 nM T47768 CUJ0N2 10331735 Ki = 1.1 nM T47768 CH14KO 10334091 EC50 = 180 nM T47768 C54WJL 10337395 Ki = 8.3 nM T47768 C63GNX 10342726 Ki = 105 nM T47768 C1VB4E 10343492 EC50 = 9 nM T47768 C3P0LR 10345440 Ki = 42 nM T47768 CJXM25 10347927 Ki = 21 nM T47768 CS3XT5 10363696 Ki = 1.04 nM T47768 C0ZF8R 10366960 IC50 = 8 nM T47768 CVQ03A 10370066 Ki > 2500 nM T47768 CFZ52M 10372345 Ki = 2.7 nM T47768 C7GK4U 10378392 Ki > 10000 nM T47768 CAYF18 10385808 Ki = 89 nM T47768 CYD30U 10387038 Ki = 7.34 nM T47768 CX2EG6 10388274 IC50 = 12110 nM T47768 CIDL30 10393594 Ki = 0.744 nM T47768 C95EWP 10395965 Ki = 90 nM T47768 C10PYA 10405782 Ki = 2040 nM T47768 CWK4O1 10406239 Ki = 0.26 nM T47768 CTA8Q0 10407144 Ki = 2.54 nM T47768 CX6ZH1 10408431 IC50 = 1.5 nM T47768 CYWF17 10412617 IC50 = 2650 nM T47768 CX4TS2 10413540 Ki = 0.11 nM T47768 C6LBC5 10415925 Ki = 630 nM T47768 CQ5HS9 10418702 Ki = 1.06 nM T47768 C7BVJ1 10428991 Ki = 0.06 nM T47768 C1U6NG 10430432 Ki = 9.4 nM T47768 CYHC38 10430819 Ki = 338.84 nM T47768 CON12X 10435156 Ki = 1.68 nM T47768 CU51WV 10440134 Ki > 4500 nM T47768 CQ4M0D 10443502 Ki = 1.8 nM T47768 C7AQ0G 10449693 IC50 = 1.9 nM T47768 CZ6I9V 10451761 IC50 = 950 nM T47768 CV14CY 10452891 IC50 = 3330 nM T47768 C0M9AN 10461299 Ki = 0.16 nM T47768 CT39OH 10462262 IC50 = 4 nM T47768 CKMN08 10475466 Ki = 398 nM T47768 CEF2O6 10478367 Ki > 10000 nM T47768 CT31DW 10479670 EC50 = 27 nM T47768 C29OZW 10484384 Ki = 42 nM T47768 CE2LD8 10486131 Ki = 35.4 nM T47768 CP72JI 10499145 IC50 > 10000 nM T47768 C1DI7F 10500922 Ki = 77 nM T47768 CGCP09 10501573 IC50 = 486 nM T47768 C90DEM 10504545 Ki = 5.9 nM T47768 C0G2QX 10508302 Ki = 52 nM T47768 CJ2BC7 10525105 IC50 = 777 nM T47768 CDGM01 10525171 IC50 = 1477 nM T47768 CT9U8L 10529438 Ki = 85.5 nM T47768 C41JWE 10546813 IC50 = 2290 nM T47768 CDK8W2 10548749 Ki = 10.9 nM T47768 CJ1TU0 10549849 IC50 = 1030 nM T47768 CKP6E2 10550601 IC50 = 597 nM T47768 CD0G5V 10552329 Ki = 1780 nM T47768 C71YXH 10553426 Ki = 5.69 nM T47768 CN4H7Z 10557001 Ki = 3200 nM T47768 CKT1L0 10569964 IC50 = 8150 nM T47768 C8E1UH 10570940 IC50 = 3570 nM T47768 CLU72B 10572649 IC50 = 2740 nM T47768 C54EOA 10572810 Ki = 16.6 nM T47768 CD9JB5 10574643 Ki = 5.9 nM T47768 C95XNB 10576543 IC50 = 4470 nM T47768 C2JU0G 10589837 IC50 = 27000 nM T47768 CQ74CO 10593778 Ki = 26 nM T47768 CT60BQ 10594839 IC50 > 10000 nM T47768 CY6D1C 10596575 IC50 = 3290 nM T47768 C2FL8C 10598391 IC50 = 620 nM T47768 C2CF1X 10598392 IC50 = 284 nM T47768 CIY19L 10600223 Ki = 203 nM T47768 C6FI2Y 10600310 Ki = 37 nM T47768 CHV5D1 10601891 Ki = 61 nM T47768 CS84IW 10618605 Ki = 12.3 nM T47768 CK96NW 10618862 IC50 = 7092 nM T47768 C62MNC 10620493 IC50 = 5064 nM T47768 CIM8S1 10620902 IC50 = 817 nM T47768 CCV14H 10642101 IC50 = 185 nM T47768 C3CHZ0 10642670 IC50 = 2980 nM T47768 C4XYH5 10644815 IC50 = 1016 nM T47768 C8ZU7I 10644995 IC50 = 2398 nM T47768 CF36MK 10645976 Ki = 26.3 nM T47768 CPC52U 10646744 Ki = 3.3 nM T47768 C10KTE 10646745 Ki = 7.5 nM T47768 CH32JY 10648307 IC50 = 6083 nM T47768 C06MRN 10651237 Ki > 4500 nM T47768 CA7Y6F 10651238 Ki > 4500 nM T47768 CC4DN0 10651452 Ki = 4500 nM T47768 CFC5R6 10668838 IC50 = 3390 nM T47768 CP5L6A 10675111 Ki > 4500 nM T47768 C84IHX 10676537 Ki > 4000 nM T47768 CA0M1N 10690216 IC50 > 10000 nM T47768 CGPT20 10692042 IC50 = 6760 nM T47768 CVS40T 10695990 IC50 = 3340 nM T47768 C3JWM0 10696939 Ki = 98.6 nM T47768 CHC1I4 10697286 Ki = 19.2 nM T47768 C5U4ZP 10713071 IC50 = 6970 nM T47768 C2RN9F 10713623 Ki = 13.3 nM T47768 C8XB3K 10714523 Ki = 31.7 nM T47768 C2W9PN 10714960 IC50 = 5050 nM T47768 C6TEF1 10717843 Ki > 2500 nM T47768 CUAC76 10718278 Ki = 10.7 nM T47768 CY9FS1 10718673 Ki > 2500 nM T47768 C3E4PH 10718848 IC50 = 5999 nM T47768 C82YCA 10719414 IC50 = 6837 nM T47768 CV8K3J 10720494 Ki = 1.6 nM T47768 CAKS63 10722490 Ki > 4500 nM T47768 CS82CN 10739828 IC50 = 2677 nM T47768 CAT04G 10741016 IC50 > 10000 nM T47768 C8RW7M 10742582 Ki = 5.16 nM T47768 CF61KY 10742765 Ki = 6.13 nM T47768 C1OBF3 10744541 Ki = 120 nM T47768 COW79X 10747714 Ki > 4500 nM T47768 CBUC04 10754185 IC50 = 6000 nM T47768 C4BJ9L 10760345 IC50 > 10000 nM T47768 CR4H2D 10760626 IC50 = 5440 nM T47768 C0PT3I 10762996 IC50 = 2222 nM T47768 CN05WO 10763594 Ki = 46.77 nM T47768 CIT9X3 10771171 Ki = 3590 nM T47768 CS1CE2 10771425 Ki = 1950 nM T47768 CDJP34 10783436 IC50 = 780 nM T47768 CB0JQ9 10785784 IC50 = 1020 nM T47768 C54YIB 10786358 IC50 = 5330 nM T47768 CSXE56 10787424 IC50 = 4130 nM T47768 CE03JT 10788324 IC50 = 9724 nM T47768 C7DVG0 10792233 Ki > 2500 nM T47768 C2O0HR 10808721 IC50 = 5980 nM T47768 C9G7LT 10809678 IC50 = 3480 nM T47768 C3ZT7Y 10810430 Ki = 1850 nM T47768 C5XWZ8 10812218 Ki = 1680 nM T47768 C2WNY5 10818843 Ki = 3280 nM T47768 C0ZOE8 10818935 Ki > 4500 nM T47768 CS3Y4G 10832076 EC50 = 31 nM T47768 CMVI50 10832445 Ki = 15.1 nM T47768 C9WI5X 10833535 IC50 = 5440 nM T47768 CPG23C 10836379 Ki = 8.4 nM T47768 C4IT2B 10837001 Ki = 2.6 nM T47768 C8S5VW 10837156 IC50 = 6186 nM T47768 COH20K 10837820 Ki > 2500 nM T47768 CFB30H 10839138 Ki = 19 nM T47768 CH53JC 10840329 Ki = 15.8 nM T47768 CN0Z1M 10841295 Ki > 4500 nM T47768 C1ZH8M 10841482 Ki > 4500 nM T47768 CFP68N 10872951 IC50 = 16.1 nM T47768 C7PR6B 10874095 IC50 = 61.8 nM T47768 CWL1K9 10874724 IC50 = 3950 nM T47768 C4ARK1 10883642 IC50 > 10000 nM T47768 C0H1TJ 10884365 IC50 > 10000 nM T47768 C9Y8OS 10884964 IC50 = 0.98 nM T47768 CRI50E 10885636 IC50 = 1470 nM T47768 CB2QL0 10885771 IC50 = 4955 nM T47768 CR2D0K 10893581 IC50 = 113 nM T47768 CE6NR5 10893607 IC50 = 421 nM T47768 C0LM2D 10893958 IC50 = 421 nM T47768 CB1HY3 10894144 IC50 = 800 nM T47768 CF61NU 10895676 IC50 = 960 nM T47768 CF3MG7 10897696 Ki = 0.17 nM T47768 CWJL70 10905740 IC50 = 6.3 nM T47768 CX65PW 10907460 IC50 = 4545 nM T47768 CQ62UO 10918307 IC50 = 179 nM T47768 CR21HO 10927114 Ki = 105 nM T47768 CT79NZ 10927276 IC50 = 1470 nM T47768 C4TSV6 10927662 Ki = 416.87 nM T47768 C1TSN4 10928037 Ki = 173.78 nM T47768 CR17TE 10928590 IC50 = 2590 nM T47768 CTN91R 10929002 IC50 > 10000 nM T47768 C9M2JE 10929207 IC50 = 735 nM T47768 C6G1ME 10930407 Ki = 0.45 nM T47768 CT5UO7 10937810 Ki = 501.19 nM T47768 CU09AV 10937901 IC50 = 1.2 nM T47768 CM0OS2 10939174 IC50 = 1730 nM T47768 C6WQ3H 10939958 IC50 = 2285 nM T47768 CS42VZ 10941213 Ki = 0.29 nM T47768 CN7XS4 10948527 IC50 = 16.7 nM T47768 CSLT97 10949380 IC50 = 2.4 nM T47768 CCUE70 10950205 IC50 > 10000 nM T47768 C9FYG3 10950562 Ki = 134.9 nM T47768 C48NDC 10950714 IC50 > 10000 nM T47768 CKR58N 10951763 Ki = 13.2 nM T47768 CHK23I 10961428 Ki = 660.69 nM T47768 CM4K7Q 10981666 IC50 = 197 nM T47768 C2HP7F 10981761 IC50 = 24.9 nM T47768 C32ZYJ 10982772 IC50 = 1.3 nM T47768 CMY56Q 10985930 Ki = 16200 nM T47768 CSZ6R2 10985963 Ki = 3100 nM T47768 C96ULE 10992239 IC50 = 458 nM T47768 CD5V9L 10992895 IC50 = 33.2 nM T47768 C91NTI 11003763 IC50 = 108 nM T47768 CJ6C9K 11003971 IC50 = 2480 nM T47768 C8Q6YE 11004121 Ki = 87.1 nM T47768 CJC9K4 11005810 IC50 = 6545 nM T47768 C3V7LT 11014751 Ki = 724.44 nM T47768 C8CP6J 11016127 IC50 = 36 nM T47768 C0VKL9 11016305 Ki = 8.86 nM T47768 C3WE6J 11024236 IC50 = 3 nM T47768 CC45BL 11025925 IC50 > 10000 nM T47768 CB7N1P 11035765 IC50 = 235 nM T47768 CUI3F2 11046929 IC50 = 16 nM T47768 C23JHR 11047568 IC50 = 1690 nM T47768 C6EBF3 11048769 IC50 > 10000 nM T47768 C57NRV 11051174 Ki > 100000 nM T47768 CL8Z9G 11058283 Ki = 5740 nM T47768 CFJG64 11059058 IC50 = 147 nM T47768 CL9Y8H 11059305 IC50 = 1235 nM T47768 C2ASJ3 11070421 Ki = 3.8 nM T47768 CG41BK 11071079 IC50 = 4015 nM T47768 CWAB48 11071778 Ki = 2.3 nM T47768 C5ZP8L 11082539 Ki = 15500 nM T47768 CS4BM0 11090195 IC50 = 94.6 nM T47768 CR0TL9 11091522 IC50 = 12.5 nM T47768 CA68BR 11091606 Ki = 33.1 nM T47768 CO08EV 11091686 IC50 > 10000 nM T47768 C6HIQ0 11092200 IC50 = 2890 nM T47768 C7WB6K 11094406 Ki = 6030 nM T47768 CONE61 11104644 Ki = 19500 nM T47768 CF0SV1 11112699 IC50 = 169 nM T47768 C7DE0U 11113605 IC50 = 3660 nM T47768 CJ25OQ 11122114 IC50 > 10000 nM T47768 C3CGB7 11123013 IC50 = 25.3 nM T47768 CM9P2I 11123816 Ki = 10.2 nM T47768 CDU0E5 11123873 Ki = 177.83 nM T47768 C6P5EL 11129476 Ki = 236 nM T47768 C9WXY1 11132954 Ki > 10000 nM T47768 CN8UZ0 11136722 Ki = 12600 nM T47768 C04HTO 11139094 IC50 = 650 nM T47768 CIL4S3 11140284 Ki = 27 nM T47768 CU6PV0 11143820 IC50 = 2 nM T47768 CP96WD 11145858 IC50 = 1.1 nM T47768 CPW06I 11146107 Ki = 2 nM T47768 C10FGZ 11149261 Ki = 312 nM T47768 C4WF6L 11152687 Ki = 17300 nM T47768 C4NAJ5 11154544 Ki = 0.28 nM T47768 CE6N5V 11157443 Ki = 7.89 nM T47768 C67ZFK 11158498 Ki = 4.7 nM T47768 CJO8S0 11163232 Ki = 48 nM T47768 C26ENL 11164004 Ki = 36.7 nM T47768 C62WBJ 11165726 Ki = 20.2 nM T47768 C6A0JS 11166820 Ki > 465 nM T47768 C26PQJ 11167140 Ki > 10000 nM T47768 C49QZC 11179386 EC50 = 1100 nM T47768 C16TCJ 11180190 Ki > 1000 nM T47768 CPQ6A8 11180584 Ki = 22.44 nM T47768 CM9TV6 11181676 Ki = 3.3 nM T47768 CLE18Z 11184156 Ki = 1080 nM T47768 CH6A1M 11184285 Ki = 40600 nM T47768 CAKZ38 11184946 IC50 = 390 nM T47768 CM6Q2S 11186913 Ki = 8.3 nM T47768 CF86JN 11188632 Ki > 5000 nM T47768 CAZ30T 11188794 Ki > 4652 nM T47768 CUBX19 11189444 IC50 = 7800 nM T47768 C90HXY 11190061 Ki = 230 nM T47768 CMRJ71 11191431 Ki = 16 nM T47768 CJL1R5 11198030 Ki = 39.7 nM T47768 CIG2Q9 11201660 Ki = 151 nM T47768 CGL3W7 11204993 Ki = 0.93 nM T47768 CS5ET8 11212373 IC50 = 24000 nM T47768 CKB01D 11212562 Ki = 6800 nM T47768 CZ4US0 11215747 Ki = 7.74 nM T47768 CK8VG1 11220535 Ki = 10.7 nM T47768 C26MVG 11223982 IC50 = 19800 nM T47768 C4QT5Y 11233481 Ki = 27.8 nM T47768 C7LD4V 11238343 Ki = 10.47 nM T47768 CA5T0Z 11238737 Ki = 29.78 nM T47768 C7DJ3L 11239327 Ki = 0.14 nM T47768 C8BO9A 11246669 Ki > 465 nM T47768 CY5S0I 11255195 Ki = 40000 nM T47768 C6V7LK 11259665 Ki = 0.664 nM T47768 C1O5ZD 11262815 Ki = 0.97 nM T47768 CF4LV5 11264459 Ki = 114 nM T47768 CCNE75 11266170 Ki = 15400 nM T47768 CCH09F 11267110 Ki = 4410 nM T47768 C9LFY6 11269707 Ki = 727 nM T47768 CD19XU 11270347 Ki = 440 nM T47768 CMI48S 11271318 Ki = 6820 nM T47768 CK90ZB 11271551 Ki = 72 nM T47768 C3G6PC 11273472 Ki = 26.28 nM T47768 CPBZ36 11274537 Ki > 5000 nM T47768 C5WYA8 11280721 Ki > 465 nM T47768 CP27SY 11283686 IC50 = 170 nM T47768 CO1HK0 11292763 Ki = 2350 nM T47768 CQ0FP3 11292970 Ki = 545 nM T47768 C59MLX 11305998 Ki = 640 nM T47768 CR4TD3 11307039 Ki = 48 nM T47768 CAWZ12 11308699 Ki = 3.3 nM T47768 CF60BC 11308721 Ki = 0.89 nM T47768 CAOJ05 11311787 Ki = 105 nM T47768 C0HCB6 11312548 Ki = 2670 nM T47768 C4FRH7 11315651 Ki > 400 nM T47768 C9A1PL 11318909 Ki = 9.83 nM T47768 CR85OX 11319221 Ki = 18.27 nM T47768 CMK6Q8 11322246 Ki = 491 nM T47768 C5DBK1 11326750 IC50 > 10000 nM T47768 CJM7R5 11327115 Ki = 210 nM T47768 CW7SN4 11329662 Ki = 53.7 nM T47768 C9D4TI 11330655 Ki = 14.67 nM T47768 CI4SY0 11333521 Ki = 17.5 nM T47768 CIS8B5 11334123 Ki = 85 nM T47768 CS1W7V 11338717 IC50 = 8040 nM T47768 CIG49E 11339827 Ki > 4652 nM T47768 C4C0OE 11341622 Ki > 10000 nM T47768 CY0SV8 11349939 Ki = 227 nM T47768 C10YKF 11351067 Ki = 7240 nM T47768 CJ9P1G 11352435 Ki = 0.5 nM T47768 C4CFD0 11358487 Ki = 422 nM T47768 CB5F8T 11359173 Ki = 5.5 nM T47768 CLT47S 11364225 Ki = 0.23 nM T47768 C73GIN 11365113 Ki = 52 nM T47768 C7QPR2 11369269 Ki = 36800 nM T47768 C6UZF7 11371415 Ki = 21.2 nM T47768 CQC4G5 11372671 IC50 = 5500 nM T47768 CA19LC 11373068 Ki > 4652 nM T47768 C9HGE1 11374952 Ki > 10000 nM T47768 CZS3E9 11376776 Ki = 3.54 nM T47768 CH50TV 11388486 Ki = 0.28 nM T47768 C5OIU1 11391288 Ki = 104 nM T47768 CR9V8F 11391721 Ki = 482 nM T47768 CT6Z0B 11393860 Ki = 38.9 nM T47768 CGO58L 11406629 IC50 = 41 nM T47768 CBJ0X5 11407510 IC50 = 3851 nM T47768 C0N5JW 11408724 Ki > 5000 nM T47768 CW0E4L 11418847 IC50 = 7180 nM T47768 CBGR89 11419799 Ki = 2980 nM T47768 C4S8GN 11421830 Ki = 14.16 nM T47768 CE8KL6 11427596 Ki = 2030 nM T47768 C85LYP 11430418 IC50 > 1000 nM T47768 CS9G3B 11430490 Ki > 4652 nM T47768 C3PD8Y 11430747 Ki > 5000 nM T47768 CY5Z6D 11434336 Ki = 1.8 nM T47768 CSZ2F1 11440849 Ki > 4652 nM T47768 C9R7AI 11444917 Ki = 17.73 nM T47768 C9KV1U 11451023 Ki = 10.6 nM T47768 C3M4ZJ 11455086 IC50 = 1.5 nM T47768 C7UDE8 11461888 Ki = 2.7 nM T47768 CKIQ83 11463791 IC50 = 11900 nM T47768 CC9TX5 11464294 IC50 = 7830 nM T47768 CMU9K5 11464846 Ki > 400 nM T47768 CMV04H 11470285 Ki = 202 nM T47768 C3T5SC 11479033 Ki = 7.89 nM T47768 C3BA5F 11480038 Ki = 2555 nM T47768 C4XU0O 11486901 Ki > 10000 nM T47768 C1LJ5U 11487063 Ki = 268 nM T47768 C5UR1M 11487946 Ki = 260 nM T47768 CA4PM8 11496383 EC50 = 120 nM T47768 CX6Q0I 11497325 Ki = 280 nM T47768 CQP65V 11503501 Ki = 18 nM T47768 CPO4E7 11507658 Ki = 13000 nM T47768 C5YIE4 11510112 IC50 = 7.8 nM T47768 C41MEV 11511090 IC50 = 4300 nM T47768 C2E7LB 11511362 Ki = 0.41 nM T47768 CZ4OM7 11516508 Ki = 68.8 nM T47768 C5LA3M 11521945 Ki = 9.5 nM T47768 CQ30PM 11525624 IC50 > 10000 nM T47768 C49XZQ 11526334 Ki = 1450 nM T47768 CB1K8W 11533999 Ki = 220 nM T47768 CF86WQ 11537712 Ki > 10000 nM T47768 CB2U5X 11540292 EC50 = 120 nM T47768 C8TZ9G 11544654 IC50 = 1300 nM T47768 CS0B4G 11544795 Ki = 288 nM T47768 COF4K0 11544824 Ki > 10000 nM T47768 CHI36N 11547640 Ki = 520 nM T47768 C3DG8U 11552010 Ki = 392 nM T47768 CHI47M 11555262 Ki = 1090 nM T47768 C2ZNA4 11558993 Ki > 10000 nM T47768 C97WYH 11559278 IC50 = 9 nM T47768 CVI52T 11561040 Ki = 4180 nM T47768 CO02FI 11562377 EC50 = 120 nM T47768 C3E4LV 11562400 Ki = 10 nM T47768 CRX48F 11581029 Ki = 58.2 nM T47768 CA35LD 11583008 Ki = 972 nM T47768 CVA8L6 11583016 IC50 > 10000 nM T47768 C3PX0F 11584092 Ki > 10000 nM T47768 CO0N2L 11591805 Ki = 30.97 nM T47768 CZA48L 11591838 Ki > 10000 nM T47768 C9GPQ8 11595485 Ki > 10000 nM T47768 C1WBQ5 11597677 IC50 > 10000 nM T47768 CY72UC 11602409 Ki = 225 nM T47768 CE4ZV5 11602862 Ki > 10000 nM T47768 C8RKH0 11619553 IC50 > 10000 nM T47768 CSYE45 11619680 EC50 = 120 nM T47768 C9WMX4 11624970 Ki = 74.4 nM T47768 C34OQC 11626062 Ki = 139 nM T47768 CM8NO4 11628123 Ki = 5660 nM T47768 C4ZD1X 11633324 IC50 > 10000 nM T47768 CZ05OM 11641014 Ki = 19 nM T47768 C2USB1 11655841 Ki = 310 nM T47768 CC1EZ6 11657075 Ki = 110 nM T47768 CQML27 11660069 Ki > 10000 nM T47768 CS91JQ 11666402 Ki > 10000 nM T47768 CXO5K2 11667199 Ki > 10000 nM T47768 C9XD2T 11677662 Ki = 0.71 nM T47768 CW7QD2 11698381 EC50 = 120 nM T47768 C19DJE 11698420 EC50 = 120 nM T47768 C79XSW 11705263 Ki = 520 nM T47768 C4ULQ7 11710187 IC50 = 1010 nM T47768 C4PXV7 11712760 EC50 = 120 nM T47768 CUG57V 11713930 Ki = 110 nM T47768 C8A2CG 11714559 Ki = 0.016 nM T47768 CC4SF3 11717551 Ki > 10000 nM T47768 COL07J 11728653 IC50 = 83.2 nM T47768 C7FSD3 11729952 IC50 = 0.65 nM T47768 C7PVL8 11730467 IC50 = 3810 nM T47768 CV3OY7 11733074 IC50 > 10000 nM T47768 CCN8E9 11742939 IC50 = 785 nM T47768 CPG15O 11743399 IC50 > 1000 nM T47768 CE0D1U 11743914 Ki = 1 nM T47768 CV8CF3 11749578 IC50 = 3920 nM T47768 CBH0Y7 11753736 Ki = 7.78 nM T47768 CFRY36 11757207 Ki = 271 nM T47768 C3F5DX 11761059 IC50 = 19.3 nM T47768 CED7I5 11761926 Ki = 275.42 nM T47768 CL6MB9 11771079 Ki = 1470 nM T47768 CEI7T9 11771732 Ki = 3.3 nM T47768 CC61WX 11773726 EC50 = 0.32 nM T47768 CX27WK 11779453 EC50 = 62 nM T47768 CJ7L9W 11784235 IC50 = 12.8 nM T47768 C1K0JF 11786990 Ki = 9.21 nM T47768 C7TLS3 11793476 IC50 = 5647 nM T47768 CJD95Z 11794240 IC50 = 5290 nM T47768 C1LJM6 11794241 IC50 = 4538 nM T47768 CG9HW8 11795019 Ki = 8.9 nM T47768 C60RKP 11796211 IC50 = 2590 nM T47768 C80ZJV 11797669 Ki = 12.8 nM T47768 C4SCZ1 11797670 Ki = 20.9 nM T47768 CX7S5D 11800732 Ki = 919 nM T47768 CJ10CQ 11803174 Ki > 4500 nM T47768 COSJ52 11811375 IC50 = 4.7 nM T47768 CN9M8E 11811722 IC50 = 83.5 nM T47768 CXY38K 11812228 IC50 > 10000 nM T47768 C8UE5W 11826819 Ki = 154.88 nM T47768 CC65TG 11827053 IC50 = 5.4 nM T47768 CS7W2V 11848793 Ki = 38 nM T47768 CHV25L 11849247 EC50 = 2.6 nM T47768 CQ6P3Y 11849249 Ki = 0.71 nM T47768 CIKN38 11849282 Ki = 0.72 nM T47768 CR47EN 11849283 Ki = 0.49 nM T47768 C7SI8L 11849284 Ki = 0.4 nM T47768 CP8QH4 11849285 EC50 = 0.04 nM T47768 C7D2TB 11849360 Ki = 0.6 nM T47768 CK2RQ0 11849361 EC50 = 0.5 nM T47768 CD39RT 11849364 EC50 = 3.8 nM T47768 CS0MC4 11950654 EC50 = 19500 nM T47768 CJ34HP 11956520 EC50 = 0.2 nM T47768 CA5ZX7 11956918 Ki = 1.1 nM T47768 CGRP40 11983337 Ki = 0.059 nM T47768 CEVH83 12041054 Ki = 8.65 nM T47768 CJP1W3 12041055 Ki = 1.54 nM T47768 C5RD1S 12041056 Ki = 0.43 nM T47768 CQ1B6S 12048050 Ki > 2930 nM T47768 C03DLA 12093958 Ki > 4500 nM T47768 CYCF29 12103026 IC50 = 1050 nM T47768 CT9KA1 12114808 Ki = 619 nM T47768 CBK43E 12114809 Ki = 1500 nM T47768 CUFP52 12149037 IC50 = 7870 nM T47768 C6IT0O 12191611 Ki = 8840 nM T47768 CYBD81 12191612 Ki = 0.65 nM T47768 CK4FE3 12298033 EC50 = 0.0051 nM T47768 CS5IZ8 12371110 Ki = 54 nM T47768 CSY9N8 12371111 Ki = 1721 nM T47768 CQI8H1 12802420 IC50 = 4.7 nM T47768 CF01LM 12986253 Ki = 0.7 nM T47768 CXF1M5 12988885 Ki > 10000 nM T47768 CNJ1Q6 13559325 Ki = 0.32 nM T47768 C06ADH 13599612 Ki = 9800 nM T47768 CAK28N 13787553 Ki = 41.7 nM T47768 C2UQX9 13911081 Ki = 410 nM T47768 C7M4BP 13911085 Ki = 833 nM T47768 CDHG39 14355117 IC50 = 7200 nM T47768 C9C5TY 14570180 Ki = 1330 nM T47768 C0UX9N 14570184 Ki = 200 nM T47768 CYW76P 14742527 Ki > 1000 nM T47768 C4EK1P 15185486 EC50 = 18400 nM T47768 CF27TQ 15384274 Ki = 2300 nM T47768 CAW1M2 15512228 Ki = 5.9 nM T47768 C30CHU 15512229 Ki = 3.981 nM T47768 C9B5OD 15512233 Ki = 398.11 nM T47768 CX6H8V 15512234 Ki = 19.95 nM T47768 CC5X0L 15512235 Ki = 10 nM T47768 CG0CS6 15512236 Ki = 39.81 nM T47768 C53KRM 15512237 Ki = 3.981 nM T47768 CLA5K8 15512238 Ki = 12.59 nM T47768 C4I5TU 15512239 Ki = 7.943 nM T47768 CSX74V 15512240 Ki = 31.62 nM T47768 CET25R 15512241 Ki = 50.12 nM T47768 C7CNY1 15512243 Ki = 25.12 nM T47768 CZA4J8 15541261 Ki = 486 nM T47768 CRM01L 15548354 Ki = 9.2 nM T47768 C1DB3A 15548355 Ki = 27.4 nM T47768 C7Q3JW 15560576 EC50 = 39.2 nM T47768 C9TYD1 15923664 Ki = 15.5 nM T47768 C75LOT 15934554 Ki = 7.9 nM T47768 CD7K0Y 15965865 IC50 = 150 nM T47768 C6DW5M 15982528 IC50 = 10000 nM T47768 C7Z8OD 15982529 IC50 = 980 nM T47768 CHO67K 15982530 IC50 = 5310 nM T47768 CV1G7O 15982660 IC50 = 840 nM T47768 CG3L8Z 15982661 IC50 = 500 nM T47768 CN64AP 15982791 IC50 = 620 nM T47768 CJ6W1T 15982933 IC50 > 10000 nM T47768 CG96OQ 15983067 IC50 = 1460 nM T47768 CV3TQ9 16006949 Ki = 0.3 nM T47768 CA5GL7 16007142 Ki = 390 nM T47768 CK3QD9 16039356 Ki = 122 nM T47768 CDR71P 16043240 IC50 = 3490 nM T47768 C3XA7E 16048783 Ki = 6.7 nM T47768 CDV05T 16048784 Ki = 5.8 nM T47768 C3O4HX 16048863 Ki = 0.29 nM T47768 CPV60X 16048864 Ki = 0.2 nM T47768 CFZI17 16048866 Ki = 2.4 nM T47768 CNDV23 16048867 Ki = 0.35 nM T47768 C9SCH7 16048936 Ki = 4 nM T47768 C6A5UL 16048937 Ki = 4.2 nM T47768 C3PO9S 16048938 Ki = 0.18 nM T47768 CJ6LM3 16048939 Ki = 2.4 nM T47768 CUQ16Z 16048940 Ki = 1.9 nM T47768 CG71OP 16048941 Ki = 0.95 nM T47768 CP23YA 16049012 Ki = 6.7 nM T47768 CQK63V 16051935 IC50 = 1 nM T47768 C6LFA8 16059781 Ki = 70 nM T47768 C4H2NO 16061455 Ki = 1175 nM T47768 C29XKY 16082873 EC50 = 20.6 nM T47768 CSK23U 16083041 Ki = 0.25 nM T47768 CR0S9Y 16087270 IC50 = 0.028 nM T47768 CSB90O 16087271 IC50 = 1.84 nM T47768 C75QOB 16087272 IC50 = 1.21 nM T47768 CP5B0A 16087273 IC50 = 0.24 nM T47768 CK8C3L 16087274 IC50 = 0.26 nM T47768 CBW82T 16087275 IC50 = 0.03 nM T47768 CFZ95P 16087276 Ki = 8.07 nM T47768 C48WDR 16087277 Ki = 3.88 nM T47768 C7V4ZB 16087278 Ki = 1.15 nM T47768 C8X5HT 16087279 IC50 = 1.45 nM T47768 CE7G1T 16087280 Ki = 1.33 nM T47768 C4B1NT 16087283 IC50 = 0.0125 nM T47768 CU1J5C 16087284 IC50 = 0.87 nM T47768 CU15KC 16087285 IC50 = 0.29 nM T47768 C30MPR 16087286 Ki = 0.86 nM T47768 CITF65 16087287 IC50 = 0.12 nM T47768 CN5KV0 16087288 IC50 = 1.27 nM T47768 C4FW9H 16087289 IC50 = 4.98 nM T47768 C2OVH1 16087290 Ki = 2.64 nM T47768 CLYD13 16094317 Ki = 430 nM T47768 C8W1BR 16094318 Ki = 110 nM T47768 C3S7GV 16094319 Ki = 73 nM T47768 CR71BM 16094320 Ki = 26 nM T47768 C6VS7F 16094321 Ki = 710 nM T47768 CV1P4O 16094322 Ki = 120 nM T47768 CZ4V9I 16094342 Ki = 110 nM T47768 CO8T5W 16094343 IC50 = 0.54 nM T47768 C0I9GV 16094344 Ki = 0.9 nM T47768 C21JYZ 16094345 Ki = 37 nM T47768 CCFS60 16094346 Ki = 940 nM T47768 CB4NE1 16094362 IC50 = 140 nM T47768 C3SZX8 16094366 IC50 = 15 nM T47768 C5RGW0 16094367 Ki = 0.98 nM T47768 CB46JH 16094368 Ki = 1.3 nM T47768 CCLO14 16094369 IC50 = 9.5 nM T47768 CUN6E1 16094370 Ki = 0.47 nM T47768 C9QI4H 16094371 Ki = 1.5 nM T47768 C90BWG 16094372 Ki = 17 nM T47768 CTY5V3 16094373 IC50 = 1.6 nM T47768 C23KIF 16094374 Ki = 4.3 nM T47768 C48EXZ 16094375 IC50 = 5.7 nM T47768 CJ7X2I 16094376 IC50 = 190 nM T47768 C9UR3E 16094377 IC50 = 6.9 nM T47768 COG76W 16094378 IC50 = 9.7 nM T47768 CBS04I 16094379 Ki = 13 nM T47768 C7AQL2 16094380 IC50 = 74 nM T47768 CMJ5H3 16094381 Ki = 3.5 nM T47768 CQ7I8F 16094382 IC50 = 80 nM T47768 CL1A7O 16094383 IC50 = 13 nM T47768 CKS40Z 16094384 IC50 = 7.5 nM T47768 CDG2M6 16094385 Ki = 15 nM T47768 C5WZF1 16094386 IC50 = 7.2 nM T47768 CYP92H 16094387 IC50 = 6.1 nM T47768 CGRX31 16094388 IC50 = 0.63 nM T47768 CO4Z1K 16094389 IC50 = 1.4 nM T47768 CH23IJ 16094390 Ki = 1.1 nM T47768 C0N6ID 16094393 Ki = 94 nM T47768 CS8L3K 16094394 Ki = 4.7 nM T47768 CX87TS 16094397 Ki = 17 nM T47768 C4RIZ1 16094408 IC50 = 52 nM T47768 C4D1UF 16094410 IC50 = 22 nM T47768 C7V1YT 16094411 IC50 = 66 nM T47768 CFRV94 16094412 Ki = 520 nM T47768 CUA2L0 16094413 IC50 = 6.7 nM T47768 C3AMW5 16094414 IC50 = 0.73 nM T47768 C6J0YV 16094415 IC50 = 13 nM T47768 CX4K0L 16094416 IC50 = 16 nM T47768 CR7AS8 16094419 IC50 = 54 nM T47768 CK98PS 16094420 IC50 = 1.1 nM T47768 C9AJK7 16094421 Ki = 3.3 nM T47768 CJ9O7S 16094422 Ki = 1600 nM T47768 CI2XK6 16094424 IC50 = 1.5 nM T47768 C6GL2A 16094425 IC50 = 2.8 nM T47768 CO4M3A 16094426 IC50 = 1.3 nM T47768 C1JBM6 16094428 Ki = 2 nM T47768 CMI74R 16094429 IC50 = 78 nM T47768 CK7N1Y 16094430 IC50 = 2 nM T47768 C8P6JV 16095099 Ki = 7 nM T47768 CI7FD0 16105558 EC50 = 82.1 nM T47768 CBL6J9 16105559 EC50 = 1.15 nM T47768 C7S6KX 16105562 EC50 = 248 nM T47768 CW17YU 16224209 Ki = 4242 nM T47768 CZ18VL 16224211 Ki = 291 nM T47768 CSG27D 16224612 Ki = 1499 nM T47768 CK5GY1 16224613 Ki = 442 nM T47768 C42GZR 16585103 EC50 = 13600 nM T47768 CZ2IS9 16660294 Ki > 10000 nM T47768 C08RXS 16665915 Ki = 500 nM T47768 CS9FW1 16665917 Ki = 1080 nM T47768 C1LX0I 16665918 Ki = 500 nM T47768 CCF0J7 16720551 EC50 = 1.7 nM T47768 C0ACW1 16720553 Ki = 22 nM T47768 CG6OD7 16720646 Ki = 3.9 nM T47768 CC4N5P 16720648 Ki = 6.7 nM T47768 CFI67Y 16720649 Ki = 0.49 nM T47768 C8GOL2 16720650 Ki = 0.37 nM T47768 CB9MZ5 16720745 Ki = 1.1 nM T47768 CAY72B 16720746 Ki = 340 nM T47768 CO84NU 16720747 Ki = 330 nM T47768 CG62NU 16720749 Ki = 0.12 nM T47768 C6W9BJ 16733371 Ki = 743 nM T47768 C8SOD5 16735664 Ki = 144 nM T47768 C4ORI6 16739256 Ki = 977 nM T47768 C1MFJ2 16747695 Ki = 163 nM T47768 C5UGV2 16748227 Ki = 4810 nM T47768 CO0XL6 16748228 Ki > 10000 nM T47768 CNEX42 16748229 Ki > 10000 nM T47768 CN4JB2 16748352 Ki = 2930 nM T47768 CJX60K 16748353 Ki > 10000 nM T47768 C5W1UD 16748354 Ki > 10000 nM T47768 C9ZD4O 16748355 Ki = 9790 nM T47768 C9TC3L 16748356 Ki = 2320 nM T47768 C68VNE 16748478 Ki = 1370 nM T47768 C6QMJ9 16756731 Ki = 400 nM T47768 C4AEU1 16756734 Ki = 59 nM T47768 C9D5RB 16756735 Ki = 45 nM T47768 C2BG6Z 16756840 Ki = 0.19 nM T47768 C0Q2OC 16756841 Ki = 54 nM T47768 C6NF5U 16756953 Ki = 33 nM T47768 CS26LH 16757050 Ki = 0.6 nM T47768 CFS39T 16757147 Ki = 8 nM T47768 C7QJW9 17379334 EC50 = 2600 nM T47768 CJNQ89 17925232 Ki > 890 nM T47768 C8AZW7 18441735 IC50 = 2700 nM T47768 C0H1TB 18545701 Ki = 265 nM T47768 C4UYA0 18607197 Ki = 1400 nM T47768 C1Y9FT 18782352 Ki = 133 nM T47768 CYUG80 18782376 Ki = 162 nM T47768 C46DPT 18782378 Ki = 130.5 nM T47768 C73DWV 18782384 Ki = 673 nM T47768 C61OBX 19881394 Ki = 325 nM T47768 C7T8JC 19958494 Ki > 10000 nM T47768 C6LI5E 19958507 Ki > 10000 nM T47768 C5BE7T 20345831 EC50 = 540 nM T47768 CIOT38 20968607 IC50 > 32000 nM T47768 CW90BF 21262767 EC50 = 102 nM T47768 C3T5HF 21509921 Ki > 10000 nM T47768 CBN84K 22065997 Ki > 10000 nM T47768 CL45HJ 22181304 Ki = 6309.57 nM T47768 CYUW32 22181436 Ki = 501.19 nM T47768 CS24KZ 22213385 Ki = 1.65 nM T47768 CHAI36 22272877 IC50 = 4400 nM T47768 CX3JY4 22273116 IC50 = 3100 nM T47768 C1W7MX 22522554 IC50 > 32000 nM T47768 C90UPB 22553442 IC50 > 32000 nM T47768 C8DF5U 22558157 Ki = 10.2 nM T47768 C0GKU4 22562137 Ki = 7.62 nM T47768 C5YZ9U 22573205 Ki = 1000 nM T47768 CJ86RS 22725091 Ki = 470 nM T47768 CD4C5N 22729898 Ki = 66.5 nM T47768 CX3O6L 22729907 Ki > 890 nM T47768 C7OL1R 22729922 Ki > 890 nM T47768 CA28YU 22729923 Ki > 890 nM T47768 CDZ19L 22733016 EC50 > 100000 nM T47768 CSP6M3 22810742 Ki = 420 nM T47768 CG60MD 22816300 Ki = 22.9 nM T47768 CL7X2U 23383556 Ki = 36 nM T47768 COHN67 23383564 Ki = 2 nM T47768 CBW20U 23435898 IC50 = 5250 nM T47768 CL45FG 23519626 IC50 = 6490 nM T47768 CDJR16 23519628 IC50 > 10000 nM T47768 CF3SU0 23519629 IC50 = 7900 nM T47768 C46ZSX 23542099 IC50 = 1190 nM T47768 CVLY78 23542106 IC50 = 2600 nM T47768 C9NI1F 23567109 Ki > 5000 nM T47768 C10UWF 23567114 Ki > 5000 nM T47768 CIPX37 23567116 Ki > 5000 nM T47768 CNH40T 23567127 Ki > 5000 nM T47768 CJD8Q6 23567134 Ki > 5000 nM T47768 C3K6HV 23594220 Ki = 1080 nM T47768 CXC6E3 23594223 Ki = 878 nM T47768 CQ93SH 23594225 Ki = 1050 nM T47768 CC5E7N 23594227 Ki = 1026 nM T47768 CG3M5J 23594230 Ki = 785 nM T47768 C5L8ZA 23594232 Ki = 319 nM T47768 C08XMZ 23594241 Ki = 1050 nM T47768 C0D5AC 23594243 Ki = 1100 nM T47768 C4JGI8 23594247 Ki = 703 nM T47768 CXN07F 23661598 Ki = 21 nM T47768 C8TEB0 23723457 EC50 = 54 nM T47768 CO5YP3 23986637 Ki = 0.32 nM T47768 CX3C6G 24735749 EC50 = 1621 nM T47768 CIW76M 24735767 EC50 = 1158 nM T47768 CB9MC8 24735827 Ki = 1761 nM T47768 C84JOU 24754997 Ki = 5.05 nM T47768 CWP85S 24776395 Ki = 476 nM T47768 CVD48X 24776396 Ki = 2075 nM T47768 C3WDL8 24776397 Ki = 540 nM T47768 CXL4R0 24776398 Ki = 1005 nM T47768 CR9I1S 24776399 Ki = 7800 nM T47768 CQDJ35 24776400 Ki = 3503 nM T47768 C6CX0Z 24776401 Ki = 1340 nM T47768 CJH18I 24776402 Ki = 6500 nM T47768 C27SGI 24776403 Ki = 1875 nM T47768 CV5IG2 24776404 Ki = 215 nM T47768 CQ70IW 24776405 Ki = 247 nM T47768 CQ2P5J 24776406 Ki = 1582 nM T47768 CYIV42 24776407 Ki = 5406 nM T47768 CWB06Z 24776408 Ki = 6755 nM T47768 C36WQO 24776409 Ki = 6139 nM T47768 CUP2C6 24776410 Ki = 5155 nM T47768 CC3W7E 24776411 Ki > 10000 nM T47768 C3N6GE 24776412 Ki = 2600 nM T47768 C2M6BR 24776413 Ki > 10000 nM T47768 CS01RL 24800107 Ki = 21 nM T47768 CL2WB0 24800108 Ki = 1.052 nM T47768 CFIS62 24822296 Ki = 0.26 nM T47768 CB4S7U 24822297 Ki = 0.43 nM T47768 CC06ON 24822298 Ki = 0.92 nM T47768 C2B3EM 24822300 Ki = 0.13 nM T47768 C1JRM9 24822458 Ki = 0.27 nM T47768 C5VYZ2 24822459 Ki = 0.38 nM T47768 CIC3L7 24822460 Ki = 1.49 nM T47768 C7O9BN 24822461 Ki = 0.64 nM T47768 C13MJI 24822630 Ki = 0.1 nM T47768 CJK3I4 24822631 Ki = 0.16 nM T47768 CW2B0R 24822632 Ki = 0.19 nM T47768 CRT19I 24822633 Ki = 0.19 nM T47768 CN6JX5 24822634 Ki = 0.21 nM T47768 CCKO91 24822798 Ki = 0.31 nM T47768 CPN52E 24822799 Ki = 0.12 nM T47768 C58EYR 24822801 Ki = 10.08 nM T47768 CBYW42 24822802 Ki = 0.12 nM T47768 CAK7O3 24822964 Ki = 0.16 nM T47768 C6R3AE 24822965 Ki = 0.43 nM T47768 CYQ27T 24824634 Ki = 0.67 nM T47768 C6TWH4 24824635 Ki = 0.05 nM T47768 CBPQ24 24824636 Ki = 0.13 nM T47768 CCY7A8 24824637 Ki = 0.18 nM T47768 C9G0CI 24824638 Ki = 0.21 nM T47768 CT0PG3 24828463 Ki = 524 nM T47768 CTZ0S2 24829369 Ki = 3.1 nM T47768 CDC91N 24839550 Ki < 10000 nM T47768 CYM02E 24847114 IC50 = 15 nM T47768 CI4W6P 24854099 Ki = 1640 nM T47768 CV6NW8 24854100 Ki = 30 nM T47768 C5ZCJ9 24854101 Ki = 7550 nM T47768 CZM9I7 24854102 Ki > 10000 nM T47768 CO7LG3 24854177 Ki = 260 nM T47768 C75WFT 24854178 Ki > 10000 nM T47768 CC5KH6 24854179 Ki = 180 nM T47768 CL06MB 24854180 Ki = 10 nM T47768 C7ED1M 24854260 Ki = 10 nM T47768 C0I4KH 24854261 Ki = 1030 nM T47768 C2ZUH5 24854262 Ki > 10000 nM T47768 CS3JT4 24854263 Ki > 10000 nM T47768 C53SWQ 24854264 Ki = 290 nM T47768 C9O5NZ 24857819 IC50 = 1900 nM T47768 CN0T1F 24857820 IC50 = 2800 nM T47768 CRUQ41 24863611 IC50 > 10000 nM T47768 CIJ83R 24873473 Ki = 0.018 nM T47768 CK61ND 24886211 Ki > 10000 nM T47768 CDR3T2 24886213 Ki > 10000 nM T47768 CNQ6I4 24894028 IC50 > 10000 nM T47768 C3C0KP 24894134 EC50 > 50000 nM T47768 CRXY84 24970014 Ki = 428 nM T47768 CT09XK 24978531 IC50 = 2690 nM T47768 CIY83H 24995848 Ki = 58.2 nM T47768 CDLW86 25001412 Ki = 190.55 nM T47768 CKNQ63 25008443 IC50 = 48 nM T47768 CQ18WG 25034086 Ki = 7 nM T47768 CTI38U 25060119 Ki = 2040 nM T47768 CU4C8F 25077980 Ki = 1740 nM T47768 C60PHW 25169521 Ki = 14 nM T47768 CV3Y7O 25169522 Ki = 450 nM T47768 CICS51 25181445 Ki = 0.1 nM T47768 CG6UT3 25181466 Ki = 0.015 nM T47768 C30VBG 25181825 IC50 > 10000 nM T47768 C4W2AK 25181826 IC50 = 5300 nM T47768 CF6RA5 25190572 Ki = 2283 nM T47768 CPK5D7 25190573 Ki = 11755 nM T47768 CON62K 25190574 Ki = 8438 nM T47768 C6S3WN 25190575 Ki = 5279 nM T47768 CKB72D 25190578 Ki = 4314 nM T47768 CZR78G 25190579 Ki = 63020 nM T47768 CF2JK0 25190580 Ki = 33120 nM T47768 CE4R2X 25190581 Ki = 13000 nM T47768 CYC6S0 25190582 Ki = 683 nM T47768 CE61QB 25190583 Ki = 483 nM T47768 C9V8MS 25190584 Ki = 726 nM T47768 C3UV5M 25190585 Ki = 886 nM T47768 CKFI42 25190586 Ki = 776 nM T47768 C5UQX3 25190587 Ki = 745 nM T47768 C5J2WE 25190588 Ki = 625 nM T47768 CX84WI 25190589 Ki = 400 nM T47768 C5RUI9 25190590 Ki = 421 nM T47768 CQY69C 25190591 Ki = 978 nM T47768 C8SEQ2 25190592 Ki = 1921 nM T47768 C5BS7N 25190593 Ki = 2546 nM T47768 CE19OU 25190594 Ki = 1376 nM T47768 CP5ID6 25190595 Ki = 1800 nM T47768 CO8E4G 25190596 Ki = 436 nM T47768 CX87HD 25190597 Ki = 683 nM T47768 CY6CV1 25190598 Ki = 29 nM T47768 CW5UP9 25190599 Ki = 146 nM T47768 C1C8VK 25190600 Ki = 167 nM T47768 CL7Q2F 25190601 Ki = 136 nM T47768 CD0H5U 25190602 Ki = 89 nM T47768 C8OWC0 25190603 Ki = 112 nM T47768 CH06YU 25190604 Ki = 28 nM T47768 CEJ25L 25190605 Ki = 26 nM T47768 CXD5R8 25190606 Ki = 122 nM T47768 CU6W8O 25190607 Ki = 142 nM T47768 CWJB54 25190608 Ki = 14 nM T47768 CMHS48 25190609 Ki = 59 nM T47768 CBL9S4 25190610 Ki = 35 nM T47768 CZ8Y6L 25190611 Ki = 37 nM T47768 CL9SN6 25190612 Ki = 69 nM T47768 C1MGY3 25190613 Ki = 96 nM T47768 CB1G6M 25190614 Ki = 120 nM T47768 CJLH27 25190615 Ki = 43 nM T47768 COE65V 25190616 Ki = 198 nM T47768 C30VGA 25190617 Ki = 64 nM T47768 CO7IV2 25190618 Ki = 239 nM T47768 C8Q7WV 25190619 Ki = 61 nM T47768 C0G4RJ 25190620 Ki = 82 nM T47768 C7X4IV 25190621 Ki = 69 nM T47768 CXG8O3 25190622 Ki = 66 nM T47768 CD5F6A 25190623 Ki = 204 nM T47768 CFUD47 25190624 Ki = 48 nM T47768 C15LIW 25190625 Ki = 102 nM T47768 C3LEW8 25190626 Ki = 139 nM T47768 CIDV61 25190627 Ki = 297 nM T47768 CAGS39 25190628 Ki = 141 nM T47768 CDS2E6 25190629 Ki = 50 nM T47768 CPW19O 25190630 Ki = 306 nM T47768 C0SBV7 25207946 Ki = 65 nM T47768 C21OJF 25207948 Ki = 11 nM T47768 C0P6CS 25207950 Ki = 20 nM T47768 CN9I8E 25208095 Ki = 3.7 nM T47768 C5OA1N 25208097 Ki = 0.59 nM T47768 C59IKP 25208099 Ki = 11 nM T47768 CUNA84 25208101 Ki = 6.3 nM T47768 C2WIG0 25208245 Ki = 45 nM T47768 CE4BI6 25208247 Ki = 151 nM T47768 CKNE16 25208249 Ki = 102 nM T47768 C57UGP 25217787 EC50 > 10000 nM T47768 C9BJD3 25232367 Ki = 0.15 nM T47768 CK0F7G 25232539 Ki = 0.14 nM T47768 CGLZ15 25232540 Ki = 0.37 nM T47768 CHG71D 25232541 Ki = 0.55 nM T47768 CGH3W8 25232542 EC50 = 0.09 nM T47768 C8E0RL 25232543 Ki = 0.11 nM T47768 CE6JP0 25232724 Ki = 0.07 nM T47768 C0OU5Y 25232725 Ki = 8.36 nM T47768 C3LHO0 25232727 Ki = 2.65 nM T47768 CO74DE 25233078 Ki = 0.12 nM T47768 CJS1L7 25233081 Ki = 0.0013 nM T47768 C1INO6 25233083 Ki = 0.1 nM T47768 C83AVG 25233258 Ki = 0.48 nM T47768 CB04CU 25235412 Ki = 777 nM T47768 CKL48U 25256790 Ki = 0.14 nM T47768 CZ2M3C 25257237 Ki = 7000 nM T47768 C9NC3W 25257431 Ki = 2.5 nM T47768 C2GH4L 25257432 Ki = 3.5 nM T47768 C0EC4L 25257433 Ki = 4.2 nM T47768 C7XY9W 25270622 IC50 > 10000 nM T47768 CBD0K9 25270623 IC50 > 10000 nM T47768 CL2Z7J 42629117 Ki = 126 nM T47768 CJ3X7R 42636619 Ki = 4900 nM T47768 C0K9TG 44138064 Ki = 0.51 nM T47768 C15NFW 44138152 Ki = 15.9 nM T47768 CL57VS 44143431 IC50 = 5600 nM T47768 C6GDL8 44143433 IC50 = 840 nM T47768 CFP9S1 44157038 Ki = 3400 nM T47768 CPQ25W 44181744 Ki = 1073 nM T47768 CX4D3R 44188273 Ki = 0.79 nM T47768 C2XE7Y 44189733 IC50 = 4500 nM T47768 CGA8R1 44189735 IC50 = 2700 nM T47768 C50FOG 44189834 IC50 = 6200 nM T47768 C2AV1K 44190762 IC50 = 1860 nM T47768 CCV87B 44235260 Ki = 1820 nM T47768 CV2NB5 44235261 Ki = 104 nM T47768 C0X3VW 44235262 Ki = 1420 nM T47768 C2HM9V 44235488 Ki = 40.2 nM T47768 CCO7H6 44235489 Ki = 713 nM T47768 CW7NH4 44235490 EC50 = 33 nM T47768 C6NIL8 44235491 Ki = 469 nM T47768 CG9QD7 44240971 Ki = 0.065 nM T47768 CR61KZ 44240972 Ki = 0.33 nM T47768 C0AL2R 44241022 Ki = 0.61 nM T47768 CK5T9S 44241023 Ki = 3.5 nM T47768 C6D0HY 44241024 Ki = 2.5 nM T47768 C5G6DN 44241123 Ki = 0.084 nM T47768 CC63QX 44247589 Ki = 123 nM T47768 CP8Q5B 44248550 Ki = 918 nM T47768 CZNM65 44248674 Ki = 596 nM T47768 C9G8KT 44248789 Ki = 1136 nM T47768 C9JBR1 44248790 Ki = 894 nM T47768 C5YV0D 44248791 Ki = 661 nM T47768 C1CZ3M 44248792 Ki = 234 nM T47768 CDG15Z 44248915 Ki = 584 nM T47768 C5I7YZ 44248916 Ki = 1684 nM T47768 C5T9AP 44248917 Ki = 8382 nM T47768 CAY83B 44248918 Ki = 891 nM T47768 CL61MJ 44248919 Ki = 5420 nM T47768 C2FLP9 44248920 Ki = 276 nM T47768 C6Q5ZF 44249045 Ki = 421 nM T47768 C0HWG8 44249046 Ki = 330 nM T47768 CHLS96 44249047 Ki = 286 nM T47768 CO4EA3 44249048 Ki = 791 nM T47768 C2SVL6 44254059 Ki = 3400 nM T47768 CVW13I 44254060 Ki = 220 nM T47768 CJW3P2 44254063 Ki = 3400 nM T47768 CZY2S1 44254585 Ki = 1800 nM T47768 CVCP62 44254956 Ki = 450 nM T47768 C8HI7P 44256416 IC50 = 22.61 nM T47768 C8DK7Z 44265058 Ki = 7500 nM T47768 CHJ15T 44265108 Ki = 1000 nM T47768 C67DCW 44268589 Ki = 11565 nM T47768 C4PG9V 44269757 IC50 = 2910 nM T47768 CW75BD 44269767 IC50 = 2100 nM T47768 CY61IX 44269822 IC50 = 9600 nM T47768 CW7C4R 44269855 IC50 > 10000 nM T47768 CUH74K 44269856 IC50 > 5000 nM T47768 CMIZ34 44269859 IC50 > 10000 nM T47768 CG93NF 44269868 IC50 > 10000 nM T47768 C35VDR 44269872 IC50 > 10000 nM T47768 C6Y8IM 44269891 IC50 = 10000 nM T47768 CM62ZD 44269901 IC50 = 1750 nM T47768 C6T9WO 44269902 IC50 > 10000 nM T47768 CQ2W3Z 44269927 IC50 > 5000 nM T47768 C2CAI8 44269932 IC50 > 10000 nM T47768 CJQI23 44269933 IC50 > 10000 nM T47768 C8AMT3 44269936 IC50 > 5000 nM T47768 C9H0AG 44269950 IC50 > 5000 nM T47768 CQ20KW 44269951 IC50 > 10000 nM T47768 C0H4SW 44269967 IC50 = 2220 nM T47768 CZ49TF 44269969 IC50 > 10000 nM T47768 CTRE60 44269980 IC50 > 10000 nM T47768 CIFJ07 44269988 IC50 = 3910 nM T47768 CWU8M4 44269994 IC50 > 10000 nM T47768 CAG2N4 44270012 IC50 = 190 nM T47768 C2CEN5 44273397 EC50 = 5.5 nM T47768 CW6P4Y 44276782 Ki = 421 nM T47768 CC2OD4 44278111 Ki > 10000 nM T47768 CRMA84 44278114 Ki > 10000 nM T47768 CF0Y4M 44278115 Ki > 10000 nM T47768 CUS04C 44279592 Ki = 0.26 nM T47768 CL70JN 44279594 Ki = 0.5 nM T47768 C3AYK9 44279686 Ki = 0.59 nM T47768 C9STZ5 44279699 Ki = 0.32 nM T47768 CN7V6X 44286598 Ki = 31.1 nM T47768 CV46BG 44286647 Ki = 1.1 nM T47768 CL72XB 44286702 Ki = 17.7 nM T47768 C6SQ3R 44286703 Ki = 31.1 nM T47768 C69JKC 44286719 Ki = 6.8 nM T47768 CY9PS5 44286720 Ki = 2.7 nM T47768 CBG62V 44286858 Ki = 21.4 nM T47768 C6NQ5U 44286870 Ki > 1000 nM T47768 C41IRN 44286883 Ki = 85.5 nM T47768 CNOB73 44286884 Ki = 392 nM T47768 C7SZ0Y 44286885 Ki = 303 nM T47768 CVAD53 44286904 Ki = 14.8 nM T47768 CW7YL3 44286905 Ki = 50.4 nM T47768 C30KQE 44286906 Ki = 34.3 nM T47768 CF7O3E 44286969 Ki = 22.8 nM T47768 CHU57Z 44287142 Ki = 38.2 nM T47768 C39XJE 44287143 Ki > 1000 nM T47768 C2Y3MA 44287144 IC50 = 894 nM T47768 CRO32K 44287168 Ki = 137 nM T47768 C09XZL 44287189 Ki = 8.8 nM T47768 C2DW5Y 44287222 Ki = 10.3 nM T47768 CJQE17 44287230 Ki = 40.5 nM T47768 CU01AP 44287231 Ki = 26.2 nM T47768 C8U5QT 44287236 Ki = 685 nM T47768 C31LOA 44287237 Ki = 56 nM T47768 CTV29Q 44287269 Ki = 33.7 nM T47768 C0RE2U 44287369 Ki > 1000 nM T47768 CO9C0E 44287381 Ki = 24 nM T47768 C83PGO 44287382 Ki = 22.7 nM T47768 CL6K5U 44287383 Ki = 395 nM T47768 CQ46MS 44287394 Ki > 1000 nM T47768 CQU8Z1 44287414 Ki = 23.2 nM T47768 C7M2FV 44287415 Ki = 173 nM T47768 CZU52X 44287483 Ki = 62.8 nM T47768 C1RE2J 44287486 Ki = 6 nM T47768 C97UNH 44287487 Ki = 5.2 nM T47768 CR6M2V 44287488 Ki = 11.7 nM T47768 CE8WC0 44288497 Ki = 700 nM T47768 C12VDA 44288499 Ki = 820 nM T47768 C6THR2 44288512 Ki = 1000 nM T47768 CJH12A 44288798 Ki = 4800 nM T47768 CVJ9M3 44288802 Ki = 17500 nM T47768 CE57CX 44288830 Ki = 20300 nM T47768 CV26NK 44288832 Ki = 650 nM T47768 C9J6GY 44288940 Ki = 475 nM T47768 C7JX2K 44288942 Ki = 425 nM T47768 C8K9AW 44288968 Ki = 5200 nM T47768 CY7S9C 44289066 Ki = 800 nM T47768 CRUP26 44289068 Ki = 760 nM T47768 C5MU4H 44289172 Ki = 10000 nM T47768 C0S9PH 44289174 Ki = 14300 nM T47768 CN46EU 44289190 Ki = 560 nM T47768 C6JH4F 44289193 Ki = 3340 nM T47768 C3BD9K 44289212 Ki = 3600 nM T47768 C2YV1Z 44289252 Ki = 4100 nM T47768 C5WE4Y 44292142 IC50 = 7220 nM T47768 C0VR9X 44292280 IC50 = 2280 nM T47768 CIEU38 44292281 IC50 = 2160 nM T47768 CARS41 44292403 IC50 = 4640 nM T47768 C2ST7W 44292414 IC50 = 142 nM T47768 C3KYZ5 44292426 IC50 = 2440 nM T47768 C2ET5R 44292437 IC50 > 10000 nM T47768 C9AF6B 44297435 Ki = 46.8 nM T47768 CNP5W1 44297519 Ki = 47.7 nM T47768 C9UY4E 44297697 Ki = 17.6 nM T47768 C8F1ST 44297727 Ki = 119 nM T47768 C4YG5R 44298841 Ki = 200 nM T47768 CF8YG9 44299258 Ki = 30 nM T47768 C7ZYM4 44299404 Ki = 504 nM T47768 CTB24D 44299841 Ki = 840 nM T47768 CT6HW3 44300146 Ki = 2.1 nM T47768 C9IL2D 44301524 Ki = 7.16 nM T47768 CG6JI1 44301701 Ki = 0.01 nM T47768 C26CLF 44302821 IC50 = 308 nM T47768 CNI7U6 44302972 IC50 = 3910 nM T47768 CL6I9X 44302973 IC50 = 1200 nM T47768 CB2H7L 44302988 IC50 = 1680 nM T47768 C28OYR 44302993 IC50 = 1100 nM T47768 C23GUZ 44303030 IC50 = 2680 nM T47768 CWM93O 44303041 IC50 = 1464 nM T47768 C4VN8H 44303094 IC50 > 10000 nM T47768 C2RTS0 44303112 IC50 > 5000 nM T47768 CGS81I 44303376 IC50 = 4840 nM T47768 CXN7F0 44303379 IC50 > 10000 nM T47768 CICN21 44303386 IC50 = 3460 nM T47768 C2L9UZ 44303682 IC50 = 4280 nM T47768 C1CI7Y 44303692 IC50 > 10000 nM T47768 CAL02W 44306565 Ki = 96 nM T47768 CT7SC8 44306566 Ki = 13.8 nM T47768 CHKQ16 44306567 Ki = 10.52 nM T47768 CR56FX 44306606 Ki = 74.73 nM T47768 CUHK45 44306640 Ki = 14.98 nM T47768 C0TKD8 44306682 Ki = 42.46 nM T47768 C5G7IS 44306729 Ki = 21.7 nM T47768 CX8UW1 44306748 Ki = 0.222 nM T47768 CTMU85 44306771 Ki = 57.74 nM T47768 C1VG3T 44306787 Ki = 3.79 nM T47768 CWT5Q7 44306866 Ki = 11.9 nM T47768 CXG6D2 44306867 Ki = 67 nM T47768 CMR0I7 44306944 Ki = 1.6 nM T47768 CEK0S4 44306977 Ki = 2.04 nM T47768 CB9P4T 44306987 Ki = 693 nM T47768 C4ZU1Q 44306988 Ki = 194 nM T47768 CUE6H5 44307017 Ki = 59 nM T47768 CZX25T 44307027 Ki = 2910 nM T47768 CMU50G 44307036 Ki = 93 nM T47768 C9SEL1 44307066 Ki = 17 nM T47768 CB74GN 44307067 Ki = 101 nM T47768 C3WRJ5 44307068 Ki = 76 nM T47768 C7K4VR 44307116 Ki = 4.8 nM T47768 CW5BN2 44307131 Ki = 294 nM T47768 CTV0Q4 44307157 Ki = 6.1 nM T47768 CRTW95 44307176 Ki = 9.58 nM T47768 CRMH14 44307182 Ki = 122 nM T47768 C0X3HL 44307191 Ki = 8 nM T47768 CW9JX4 44307198 Ki = 0.654 nM T47768 CM6J0K 44307210 Ki = 21.7 nM T47768 CY1H2U 44307211 Ki = 13.48 nM T47768 CQ2HL0 44307228 Ki = 8.72 nM T47768 C82AYR 44307326 Ki = 2.52 nM T47768 CTX9O8 44307330 Ki = 0.14 nM T47768 CI8XV3 44307356 Ki = 417 nM T47768 CC7F4Q 44307381 Ki = 61 nM T47768 C5G2VA 44307382 Ki = 84 nM T47768 CCN57J 44307428 Ki = 6.77 nM T47768 C0GJT5 44311043 Ki = 4 nM T47768 C2GE8X 44311351 Ki = 0.7 nM T47768 CV9X4Q 44311893 Ki = 5.33 nM T47768 CLX5V8 44312109 Ki = 17.4 nM T47768 CK6IY4 44315305 Ki = 19.95 nM T47768 CM0G8A 44324324 Ki = 3200 nM T47768 CALT96 44324339 Ki = 1700 nM T47768 C2Y4SJ 44324361 Ki = 5700 nM T47768 CT39YA 44324362 Ki = 5250 nM T47768 CY9BC0 44326368 IC50 = 1.6 nM T47768 C0BR8P 44326371 IC50 = 1.3 nM T47768 C0FUD3 44326372 IC50 = 2 nM T47768 C7F8TX 44326413 IC50 = 0.88 nM T47768 CE9W0C 44326414 IC50 = 5.9 nM T47768 CE69ON 44326415 IC50 = 0.74 nM T47768 CY1ML0 44326426 IC50 = 8.3 nM T47768 CR8K3D 44326480 Ki = 22.32 nM T47768 C5NHT1 44329096 Ki > 6000 nM T47768 CV57DK 44329162 Ki = 140 nM T47768 C8ABT2 44329206 Ki > 6000 nM T47768 CH46CQ 44329417 Ki = 4500 nM T47768 CV91DR 44329508 Ki > 6000 nM T47768 CL3B0J 44329509 Ki = 2000 nM T47768 C1LOP6 44329524 Ki > 6000 nM T47768 C2JOC8 44329698 Ki = 1300 nM T47768 CV90JY 44329722 Ki = 7900 nM T47768 C9YU3Z 44329726 Ki > 6000 nM T47768 COE92S 44329727 Ki > 6000 nM T47768 COR3H8 44329728 Ki > 6000 nM T47768 CAS38O 44332117 Ki = 16.4 nM T47768 CR0UZ9 44333058 Ki = 1.97 nM T47768 C26IAM 44336365 Ki = 0.08 nM T47768 CJ4WL1 44336602 Ki = 0.79 nM T47768 CM3K9Y 44336603 Ki = 204 nM T47768 CW14ZR 44336650 Ki = 135 nM T47768 CXC23A 44336684 Ki = 163 nM T47768 CXUR84 44336767 Ki = 1056 nM T47768 CZ0E6U 44336783 Ki = 1151 nM T47768 CGZ9N2 44336905 Ki = 1766 nM T47768 CYMH75 44337108 Ki = 7159 nM T47768 CJ0I6Q 44337123 Ki = 4317 nM T47768 CPOX86 44337129 Ki = 5401 nM T47768 CT78UG 44337131 Ki = 516 nM T47768 CO8Y5G 44337163 Ki = 2248 nM T47768 CBJ01F 44337212 Ki = 3975 nM T47768 C8IJM5 44337229 Ki = 1599 nM T47768 C97YKG 44337230 Ki = 10620 nM T47768 C3B4WO 44337231 Ki = 801 nM T47768 CU8IY3 44337232 Ki = 2502 nM T47768 C3M0QX 44337249 Ki = 4705 nM T47768 C0MJL2 44337252 Ki = 9666 nM T47768 CB85KA 44337351 Ki = 7217 nM T47768 CI13YG 44337357 Ki = 586 nM T47768 CW2FZ7 44337362 Ki = 865 nM T47768 CJ08FM 44337379 Ki = 1815 nM T47768 CIP87K 44337437 Ki = 1494 nM T47768 CR62KO 44337452 Ki = 6015 nM T47768 C9CIP3 44337459 Ki = 3452 nM T47768 CFA2Q7 44337460 Ki = 2176 nM T47768 CF96JK 44337473 Ki = 4130 nM T47768 CX87AS 44337513 Ki = 2148 nM T47768 CP1VN3 44337550 Ki = 1591 nM T47768 CZ02BO 44337551 Ki = 1939 nM T47768 C4AIE7 44337613 Ki = 0.43 nM T47768 CHB64V 44337616 Ki = 13.58 nM T47768 C35PQC 44337617 Ki = 4.8 nM T47768 CKZ03N 44337618 Ki = 37.64 nM T47768 C7A9FQ 44337642 Ki = 254 nM T47768 C6AVW4 44337643 Ki = 4.64 nM T47768 C8OFG5 44337644 Ki = 37.05 nM T47768 C59RIN 44337645 Ki = 330 nM T47768 C18MWY 44337673 Ki = 22.97 nM T47768 CI8AT5 44337683 Ki = 4.54 nM T47768 C0J9UR 44337749 Ki = 43.95 nM T47768 CJTU61 44337750 Ki = 61.91 nM T47768 CMGC86 44337764 Ki = 26.35 nM T47768 CI48SV 44337765 Ki = 31.59 nM T47768 CVP73N 44337783 Ki = 13.48 nM T47768 C7Q4HS 44337789 Ki = 6.3 nM T47768 CP4A0K 44337800 Ki = 13.4 nM T47768 C64JKH 44337822 Ki = 56.62 nM T47768 C20HGO 44337823 Ki = 25.29 nM T47768 C40VWE 44337830 Ki = 40.79 nM T47768 C3QGP4 44337831 Ki = 47.4 nM T47768 CHVG85 44337832 Ki = 23.53 nM T47768 CS57JZ 44337839 Ki = 122 nM T47768 CS9Z1O 44339374 Ki = 4 nM T47768 CF08RA 44339398 Ki > 10000 nM T47768 C9CIL3 44339409 EC50 = 9.8 nM T47768 CFNR91 44339423 Ki = 8 nM T47768 CW56BK 44339424 Ki = 36 nM T47768 C4POK5 44339425 Ki = 46 nM T47768 C7HIP9 44339463 Ki = 2.5 nM T47768 CF1HE6 44339472 EC50 > 10000 nM T47768 CFRJ92 44339475 EC50 = 3.47 nM T47768 C73QPW 44339504 Ki = 626 nM T47768 C68ZSO 44339521 EC50 = 1.97 nM T47768 C7GRF4 44339525 Ki = 104 nM T47768 CX93QM 44339562 Ki = 192 nM T47768 CO9IF8 44339563 Ki = 0.492 nM T47768 C7E4MS 44339576 Ki = 124 nM T47768 C2PDT6 44339596 Ki = 113 nM T47768 C34DEN 44339684 Ki = 19 nM T47768 CO3C7M 44339695 Ki = 21 nM T47768 CM42BN 44341722 Ki = 3.75 nM T47768 CND5T9 44341920 Ki = 7.32 nM T47768 CM4NE8 44342057 IC50 = 6.3 nM T47768 C6BX2A 44342141 IC50 = 2590 nM T47768 CD9ZS8 44342270 IC50 = 16 nM T47768 C4N6GE 44342597 Ki = 183 nM T47768 C0Z9DY 44342598 Ki = 59 nM T47768 CSZ34A 44342661 Ki = 27 nM T47768 CJVN97 44342684 Ki = 126 nM T47768 CP97HW 44342724 Ki = 259 nM T47768 C2EQZ1 44342741 Ki = 776 nM T47768 CYTQ61 44342743 Ki = 318 nM T47768 C0IJN7 44342746 Ki = 160 nM T47768 CQ5B8R 44342747 Ki = 997 nM T47768 CW5RB3 44342753 Ki = 4186 nM T47768 C1LQR9 44342754 Ki = 1378 nM T47768 CD3F2N 44342792 Ki = 1241 nM T47768 CC1X5F 44342793 Ki = 943 nM T47768 C46PTB 44342843 Ki = 756 nM T47768 CNO76C 44342910 Ki = 4.2 nM T47768 C5NQP9 44342911 Ki = 1.5 nM T47768 CNG79I 44342912 Ki = 15 nM T47768 CLC0Z1 44342925 Ki = 39 nM T47768 C74GDW 44342933 Ki = 3.4 nM T47768 CG1X6K 44342934 Ki = 16 nM T47768 CTR31B 44343016 Ki = 0.29 nM T47768 CA94RF 44343030 Ki = 13.6 nM T47768 C0YV2K 44346065 Ki = 0.12 nM T47768 C0JWA6 44348797 IC50 = 20286 nM T47768 CPV8R3 44349947 Ki = 3 nM T47768 C4HYP6 44355590 Ki = 5200 nM T47768 CL2JI8 44355639 IC50 = 720 nM T47768 CCI68O 44355640 IC50 = 4300 nM T47768 CVO2G3 44355745 Ki = 5.7 nM T47768 CMS4H1 44355747 Ki = 25 nM T47768 C8VW0Y 44355787 Ki = 136 nM T47768 C4YF9A 44356081 IC50 = 77000 nM T47768 CX8OV0 44358749 IC50 = 16 nM T47768 C1CNB6 44358751 Ki = 850 nM T47768 C9QT7R 44358763 IC50 = 24 nM T47768 CZRQ16 44358764 Ki = 150 nM T47768 CT6IW3 44358829 Ki = 5.5 nM T47768 CR7B2P 44358857 Ki = 5.3 nM T47768 C1UXN9 44358875 Ki = 5 nM T47768 C84JQO 44358880 Ki = 0.5 nM T47768 CYK75T 44358889 Ki = 3.2 nM T47768 CD2KB4 44358890 Ki = 3.1 nM T47768 CG7H8O 44358892 Ki = 1.7 nM T47768 CTE6H7 44358901 Ki = 1200 nM T47768 C5R1NH 44358904 Ki = 9.7 nM T47768 CA21BS 44358922 Ki = 8.8 nM T47768 CI0Q7R 44358923 Ki = 8.3 nM T47768 C1JUA9 44358924 Ki = 8 nM T47768 CYK1G5 44358967 Ki = 6.2 nM T47768 C0X9FD 44358968 Ki = 53 nM T47768 CG68ZO 44358969 IC50 = 2.1 nM T47768 CH65DU 44358987 Ki = 69 nM T47768 CHY6F1 44359130 Ki = 29 nM T47768 C8H1FC 44359131 Ki = 16 nM T47768 CP58ZU 44359139 Ki = 15 nM T47768 CYN3L7 44359140 Ki = 13 nM T47768 CWFQ58 44363688 Ki = 433 nM T47768 CST17U 44363907 Ki = 23 nM T47768 CZTA92 44363923 Ki = 37 nM T47768 CHGO26 44363938 Ki = 477 nM T47768 CD18TR 44366689 Ki = 2700 nM T47768 CYL95J 44366690 Ki = 496 nM T47768 C7IFR8 44366822 Ki = 53 nM T47768 CL1JV2 44366823 Ki = 75 nM T47768 COEC43 44367007 Ki > 10000 nM T47768 CTY04M 44367017 Ki = 21 nM T47768 CT71JB 44367028 EC50 = 34 nM T47768 C30QSI 44367136 Ki = 16.8 nM T47768 C8IZ2L 44367182 Ki = 49.5 nM T47768 CRO21Y 44367308 Ki = 40.1 nM T47768 C8BX2S 44367339 Ki = 52.7 nM T47768 CF5Q6M 44368739 Ki = 1.97 nM T47768 C7EMY8 44368740 Ki = 1.12 nM T47768 C9XK2F 44374175 Ki = 1.2 nM T47768 CF9Z8Q 44374177 Ki = 0.24 nM T47768 C13FDT 44374197 Ki = 1.2 nM T47768 CRZ03M 44374199 Ki = 0.42 nM T47768 CXM2W1 44374294 Ki = 1.6 nM T47768 C95JYL 44374319 Ki = 0.69 nM T47768 CBPG98 44374358 Ki = 0.72 nM T47768 C6AJ1E 44374448 Ki = 0.64 nM T47768 CNI91A 44374450 Ki = 0.37 nM T47768 C7XG9B 44380504 Ki = 0.6 nM T47768 CL89XO 44380683 Ki > 10000 nM T47768 CCX1K8 44380752 Ki = 3350 nM T47768 CE0C5H 44380980 EC50 = 21 nM T47768 CT84GR 44380994 EC50 = 22 nM T47768 CV6E7J 44381061 Ki > 10000 nM T47768 CK8SV3 44381244 Ki = 18 nM T47768 CAL7O1 44390336 Ki = 8.7 nM T47768 C65UZW 44390346 Ki = 5.4 nM T47768 C5I7AN 44390989 Ki = 58 nM T47768 C2W7BJ 44391023 Ki = 410 nM T47768 CF49QH 44391052 Ki = 38 nM T47768 C7A8DM 44391062 Ki = 65 nM T47768 CTA04B 44391063 Ki = 103 nM T47768 C1WGX6 44391067 Ki = 103 nM T47768 C8Y7OV 44391069 Ki = 196 nM T47768 CY7OH0 44391079 Ki = 21 nM T47768 CPZ7L8 44391081 Ki = 166 nM T47768 CR5TN7 44391092 Ki = 23 nM T47768 C2DB4N 44391093 Ki = 355 nM T47768 CO2T5M 44391094 Ki = 47 nM T47768 CL79EO 44391099 Ki = 118 nM T47768 C3HTZ1 44391102 Ki = 477 nM T47768 CW76ZY 44391103 Ki = 24 nM T47768 CN1LD9 44391104 Ki = 114 nM T47768 CD3QV8 44391111 Ki = 45 nM T47768 CK2HV1 44391119 Ki = 20 nM T47768 C8RDV5 44391124 Ki = 58 nM T47768 C1UDL9 44391133 Ki = 27 nM T47768 CSV6X2 44391134 Ki = 67 nM T47768 CJ9MX1 44391137 Ki = 102 nM T47768 C18SDI 44391138 Ki = 56 nM T47768 C6ZF9E 44391155 Ki = 16.7 nM T47768 CY6T4F 44391156 Ki = 88 nM T47768 CJB0U8 44391157 Ki = 62 nM T47768 C5ZFX2 44394283 Ki = 188 nM T47768 COB70L 44394284 Ki = 73 nM T47768 C6DB4X 44394324 Ki = 91.7 nM T47768 C2OV9B 44394344 Ki = 660 nM T47768 CCR2U1 44394375 Ki = 13 nM T47768 CQ2O6J 44394381 Ki = 92 nM T47768 CTJ2I9 44394405 Ki = 289 nM T47768 CLFU54 44394419 Ki = 1376 nM T47768 C0A1OW 44394487 Ki = 106 nM T47768 CRCV49 44394559 Ki = 294 nM T47768 C3YD8C 44395259 Ki = 8128 nM T47768 CR8AF5 44395265 Ki = 331 nM T47768 CI7GR3 44395286 Ki = 0.3 nM T47768 CLB5E3 44395291 Ki = 489 nM T47768 CEX0W2 44395306 Ki = 0.23 nM T47768 C69ACH 44395319 Ki = 1461 nM T47768 CQO0Y5 44395366 Ki > 10000 nM T47768 C0FUP2 44395387 Ki > 10000 nM T47768 C06LKH 44395410 Ki = 37 nM T47768 CL6WV3 44398138 Ki > 10000 nM T47768 CJ98TY 44398175 Ki = 73 nM T47768 C56JOK 44399274 Ki = 1240 nM T47768 CPSF28 44399379 Ki = 2300 nM T47768 CC1UY9 44399493 Ki = 478 nM T47768 C4XEQ2 44399584 Ki = 570 nM T47768 CR0G7H 44399648 Ki = 1062 nM T47768 CT2YO6 44399674 Ki = 1900 nM T47768 CMA91N 44399675 Ki = 74 nM T47768 CXR91I 44401402 Ki = 11 nM T47768 CQRZ78 44401457 Ki = 0.13 nM T47768 C3Y4MD 44401653 Ki = 17 nM T47768 C1B4QL 44403095 Ki > 10000 nM T47768 C1YL7Z 44403098 Ki > 10000 nM T47768 CFV98A 44403101 Ki > 10000 nM T47768 C6OY9S 44403102 Ki > 10000 nM T47768 CH4SX6 44403105 Ki > 10000 nM T47768 C12FIH 44403106 Ki > 10000 nM T47768 CIP16C 44403937 Ki = 33 nM T47768 C4LKC1 44404394 Ki > 10000 nM T47768 C3EJ4G 44404396 Ki > 10000 nM T47768 C7GP1E 44404646 IC50 = 1690 nM T47768 CILB28 44404652 IC50 = 1110 nM T47768 CA58SU 44404670 IC50 = 960 nM T47768 C83PCH 44404679 IC50 = 3550 nM T47768 CU0YX9 44404684 IC50 = 1610 nM T47768 CEJ7F8 44404689 IC50 > 10000 nM T47768 CODG94 44404695 IC50 = 6470 nM T47768 CD79WM 44404698 IC50 = 4280 nM T47768 C0BED6 44404699 IC50 = 480 nM T47768 C2NHS0 44404707 IC50 > 10000 nM T47768 CNX5T8 44404731 IC50 = 1410 nM T47768 CE41AD 44405138 Ki > 5000 nM T47768 CN0G4K 44405139 Ki > 5000 nM T47768 CE81GQ 44405140 Ki > 5000 nM T47768 CU02RP 44405141 Ki > 5000 nM T47768 CUIG59 44405142 Ki > 5000 nM T47768 CA2B3X 44405144 Ki > 5000 nM T47768 C1UZE3 44405145 Ki > 5000 nM T47768 CYX81F 44405161 Ki > 5000 nM T47768 CHU8N9 44405164 Ki > 5000 nM T47768 C0AXJ5 44405165 Ki > 5000 nM T47768 CV5Y3I 44405172 Ki > 5000 nM T47768 CM05NC 44406109 Ki > 4652 nM T47768 CA0RM2 44406110 Ki > 4652 nM T47768 C2T6WY 44406111 Ki = 2520 nM T47768 C5P9NO 44406128 Ki > 4652 nM T47768 CI2C5K 44406161 Ki > 4652 nM T47768 CRL3P8 44406171 Ki > 4652 nM T47768 CQ2D6B 44406177 Ki = 1206 nM T47768 CALG92 44406185 Ki > 4652 nM T47768 C7WQ5V 44406186 Ki = 3246 nM T47768 CBH5G9 44406215 Ki = 1417 nM T47768 CRI8L5 44406219 Ki = 497 nM T47768 CUH65A 44406224 Ki > 4652 nM T47768 CF61YM 44406225 Ki = 1385 nM T47768 CKS9V8 44406273 Ki = 428 nM T47768 CS7KQ8 44406280 Ki > 465 nM T47768 CLE5R9 44406285 Ki > 4652 nM T47768 CZFM30 44406286 Ki > 4652 nM T47768 C57ADM 44406306 Ki > 465 nM T47768 CVX84Y 44406350 Ki > 4652 nM T47768 C0C2BN 44406353 Ki = 235 nM T47768 CJ6H4U 44406370 Ki > 4652 nM T47768 C79UVP 44406376 Ki > 4652 nM T47768 CW9QG2 44406457 IC50 = 3000 nM T47768 CGN73V 44406458 IC50 = 1000 nM T47768 C0J7IK 44406489 IC50 = 150 nM T47768 C5TIM4 44406497 IC50 = 3600 nM T47768 CBUR32 44406503 IC50 = 4000 nM T47768 C17FYG 44406538 IC50 = 2700 nM T47768 C07CNE 44406539 IC50 = 2500 nM T47768 C5DGV2 44406540 IC50 = 1090 nM T47768 C9Z0ET 44406541 IC50 = 2200 nM T47768 C1L8CG 44406543 IC50 = 2400 nM T47768 CP1OZ6 44406544 IC50 = 4400 nM T47768 CS04TK 44406550 IC50 = 2170 nM T47768 C8HRC9 44406551 IC50 = 1420 nM T47768 CSPE30 44406557 IC50 = 1800 nM T47768 CZPS59 44406568 IC50 = 0.6 nM T47768 CD7Y0Z 44406585 IC50 = 2200 nM T47768 CC15BY 44406587 IC50 = 3700 nM T47768 C1IM9R 44406603 IC50 = 4000 nM T47768 C3VE8N 44406604 IC50 = 260 nM T47768 CL3EO9 44406605 IC50 = 130 nM T47768 CCI5Z1 44406618 IC50 = 540 nM T47768 C7ES2W 44406621 IC50 = 1600 nM T47768 C0SKT9 44406641 IC50 = 3200 nM T47768 C4RJY2 44406656 Ki = 130 nM T47768 CSMQ84 44406657 Ki = 0.67 nM T47768 CSF2Y6 44406658 Ki = 0.65 nM T47768 C2KBP7 44406663 Ki = 0.01 nM T47768 C38ABN 44406682 IC50 = 5300 nM T47768 CZ65PF 44406685 IC50 = 2500 nM T47768 C3SEN7 44406695 Ki = 2.8 nM T47768 C2MR7W 44406696 Ki = 0.71 nM T47768 C4LA2U 44406703 Ki = 2.2 nM T47768 COG8U3 44406710 Ki = 3.3 nM T47768 CZC51G 44406712 Ki = 5.7 nM T47768 CPO9T5 44406713 Ki = 13 nM T47768 CWY76P 44406719 IC50 = 230 nM T47768 CRE4Q9 44406723 Ki = 0.22 nM T47768 C4N1MC 44406724 Ki = 0.44 nM T47768 CB30EK 44406732 Ki = 0.34 nM T47768 CVER25 44407299 Ki = 75 nM T47768 C9AU3C 44407301 IC50 = 15 nM T47768 CVP98E 44407305 Ki = 280 nM T47768 C4J3VF 44407309 IC50 = 280 nM T47768 C3NG6O 44407310 Ki = 160 nM T47768 C7YM3D 44407311 IC50 = 16 nM T47768 C2QNC5 44407312 IC50 = 170 nM T47768 C3DQ8W 44407313 IC50 = 100 nM T47768 CQ9X8L 44407315 Ki = 15 nM T47768 CX82DC 44407316 Ki = 230 nM T47768 CD9R7C 44407317 Ki = 560 nM T47768 CY3EH0 44407318 IC50 = 170 nM T47768 CU6D4P 44407323 Ki = 270 nM T47768 CJ51HQ 44407324 Ki = 110 nM T47768 C2I8RZ 44407329 IC50 = 390 nM T47768 CW89MA 44407330 IC50 = 130 nM T47768 CTLY61 44407348 Ki = 59 nM T47768 CE9K1V 44407351 Ki > 1000 nM T47768 CY8R2X 44407359 IC50 = 320 nM T47768 C69OZA 44407360 IC50 = 290 nM T47768 CB16YW 44407361 IC50 = 210 nM T47768 C2P4ZH 44407364 IC50 = 39 nM T47768 CG87PW 44409290 Ki > 1000 nM T47768 C59XVU 44411613 Ki > 10000 nM T47768 CYE4D3 44411762 Ki > 10000 nM T47768 CMG79P 44411790 Ki > 10000 nM T47768 CS0ZC2 44411794 Ki = 430 nM T47768 CDK08M 44411860 Ki > 10000 nM T47768 C52WZH 44413231 Ki > 10000 nM T47768 CFJ64A 44413232 Ki = 2700 nM T47768 CNFC81 44413248 Ki > 5000 nM T47768 C0V4FI 44413286 Ki = 2000 nM T47768 CS7BI8 44413301 Ki = 900 nM T47768 C1NGS0 44413314 Ki = 530 nM T47768 C5J0BU 44413315 Ki > 5000 nM T47768 CH7E1C 44413329 Ki > 5000 nM T47768 C1OQ0L 44413330 Ki = 170 nM T47768 CKV5S0 44413361 Ki = 900 nM T47768 C5PHK7 44413362 Ki = 760 nM T47768 CSQZ28 44413379 Ki = 500 nM T47768 CCU2B5 44413384 Ki = 430 nM T47768 CD5SZ9 44413385 Ki = 260 nM T47768 C7GE2K 44413395 Ki > 5000 nM T47768 CCK6Y5 44413396 Ki = 4140 nM T47768 C0FL8K 44413401 Ki > 5000 nM T47768 C6J3HP 44413402 Ki > 5000 nM T47768 CB2OJ9 44413408 Ki > 5000 nM T47768 C82VJB 44413413 Ki = 330 nM T47768 CP31JV 44413414 Ki = 340 nM T47768 C98OQG 44413423 Ki = 880 nM T47768 CH0DS7 44413441 Ki = 1360 nM T47768 CLSK72 44413442 Ki = 260 nM T47768 C3J4VM 44414717 IC50 = 1870 nM T47768 C6O2VL 44414730 IC50 > 10000 nM T47768 C7N9AR 44414747 IC50 = 5480 nM T47768 CRCQ06 44414830 IC50 = 1550 nM T47768 C1PK7O 44414844 IC50 > 10000 nM T47768 C5Z9VE 44414845 IC50 = 6700 nM T47768 C4LI9Q 44414865 IC50 = 1090 nM T47768 CWR4S6 44414876 IC50 = 3030 nM T47768 CU65WM 44415621 Ki = 18 nM T47768 C1MO6K 44415676 Ki = 6.4 nM T47768 C7U8LB 44415720 Ki = 27 nM T47768 C1UT9Q 44415832 Ki = 3.1 nM T47768 CUF36X 44417374 Ki = 0.32 nM T47768 CFJC63 44417384 Ki = 0.7 nM T47768 C72HIJ 44421393 Ki = 7.6 nM T47768 C0M1LF 44421396 Ki = 8.75 nM T47768 CI12ZC 44421399 Ki = 5.06 nM T47768 COM3F5 44421400 EC50 = 2.51 nM T47768 C2L4MW 44421401 Ki = 5.39 nM T47768 CKA1J2 44421403 Ki = 18.5 nM T47768 C5S4EC 44421406 Ki = 7.46 nM T47768 CW6I0V 44421407 Ki = 25.2 nM T47768 CN6E4Q 44421408 Ki = 25.8 nM T47768 CLEH29 44421409 Ki = 88.9 nM T47768 C4ZXO2 44421412 Ki = 17.9 nM T47768 C5K6YB 44421422 Ki = 15.4 nM T47768 C9ACE6 44422807 Ki = 0.46 nM T47768 C2IE1L 44422808 Ki = 0.29 nM T47768 C0Q8TZ 44425152 Ki > 10000 nM T47768 C4NWJ9 44425154 Ki > 10000 nM T47768 CYQ28K 44425156 Ki = 1530 nM T47768 C10OMS 44426811 Ki = 125 nM T47768 C49KAS 44426813 Ki = 787 nM T47768 CJ5FC0 44426816 Ki = 780 nM T47768 C4TFP1 44426818 Ki = 59810 nM T47768 CP5V8D 44426821 Ki = 3736 nM T47768 C5L4SE 44426822 Ki = 9324 nM T47768 C36SCP 44426823 Ki = 819 nM T47768 C72RXV 44426824 Ki = 405 nM T47768 C0S5TE 44426829 Ki = 127 nM T47768 CL1EG2 44426830 Ki = 714 nM T47768 CBFY73 44426831 Ki = 1207 nM T47768 CFO9Q6 44426832 Ki = 9 nM T47768 C2NFA4 44426833 Ki = 201 nM T47768 COJ48Z 44426834 Ki = 793 nM T47768 CUD42S 44426835 Ki = 177 nM T47768 CKJ90O 44426836 Ki = 170 nM T47768 CZ4R6J 44426837 Ki = 2449 nM T47768 CPDE73 44426838 Ki = 120 nM T47768 C53JGK 44426839 Ki = 2864 nM T47768 C7IJY0 44426840 Ki = 148 nM T47768 CJB90W 44426841 Ki = 183 nM T47768 CK3B6E 44426843 Ki = 843 nM T47768 CD3TB8 44426844 Ki = 843 nM T47768 CFY3A6 44427433 Ki = 7 nM T47768 C0M4EP 44427434 Ki = 0.19 nM T47768 CT2Z8J 44429058 Ki = 150 nM T47768 CQ87UY 44429059 Ki = 40 nM T47768 CF5OJ0 44430021 Ki = 8382 nM T47768 CUQ95Y 44430022 Ki = 186 nM T47768 CZA0E6 44430023 Ki = 125 nM T47768 CWX67P 44430033 Ki = 756 nM T47768 C40BHT 44430038 Ki = 2 nM T47768 C1QXR6 44430040 Ki = 28 nM T47768 CS6Y5Z 44430042 Ki = 72 nM T47768 C4CHV5 44430043 Ki = 72 nM T47768 CX9P5R 44430044 Ki = 190 nM T47768 CA51JN 44430045 Ki = 502 nM T47768 C2G9HQ 44430046 Ki = 3085 nM T47768 C8PI4A 44430047 Ki = 616 nM T47768 CL1N4D 44430048 Ki = 452 nM T47768 C0AYM6 44430049 Ki = 181 nM T47768 CMJT74 44430050 Ki = 167 nM T47768 C4ZG6A 44430079 Ki = 198 nM T47768 CSNQ43 44430080 Ki = 304 nM T47768 CXV9J7 44430081 Ki = 120 nM T47768 CFHY18 44430083 Ki = 145 nM T47768 C6SBE1 44430084 Ki = 190 nM T47768 CXZ2D3 44430085 Ki = 351 nM T47768 CI4X3Z 44430087 Ki = 353 nM T47768 C15KTO 44432560 Ki > 465 nM T47768 C47USK 44432561 Ki > 465 nM T47768 C9KQE6 44432562 Ki > 465 nM T47768 C8W2RQ 44432563 Ki > 465 nM T47768 CT4P1M 44432564 Ki > 4652 nM T47768 CDP72X 44432565 Ki > 465 nM T47768 CJQC39 44432566 Ki > 4652 nM T47768 CHNQ16 44432567 Ki > 465 nM T47768 C6TD1E 44432583 Ki > 465 nM T47768 CQ4X2F 44432589 Ki > 4652 nM T47768 C97UQG 44432591 Ki > 4652 nM T47768 CJN2O9 44432597 Ki > 465 nM T47768 CM3P1O 44432599 Ki > 465 nM T47768 C37YLC 44432606 Ki > 465 nM T47768 CA9S4M 44432608 Ki > 465 nM T47768 CG7KL2 44432609 Ki > 4652 nM T47768 CLQH28 44432610 Ki > 4652 nM T47768 C3W6AY 44432611 Ki > 465 nM T47768 CU8F0D 44432613 Ki > 465 nM T47768 CC15LP 44432614 Ki > 465 nM T47768 COM06U 44432615 Ki > 465 nM T47768 CG69US 44432616 Ki > 465 nM T47768 CF02PQ 44433159 Ki > 465 nM T47768 C34OTB 44433399 Ki = 13 nM T47768 CT4QL9 44433400 Ki = 20 nM T47768 CO08LU 44433401 Ki = 34 nM T47768 CC5G2Y 44433402 Ki = 4.3 nM T47768 CJ20NZ 44434062 Ki = 179 nM T47768 CF78VR 44434063 Ki = 15.95 nM T47768 C38NOM 44434064 Ki = 185 nM T47768 CT8QH4 44434065 Ki = 231.59 nM T47768 CTM38X 44434066 Ki > 3333 nM T47768 CMT4U1 44434067 Ki = 10.09 nM T47768 CF0V8Z 44434068 Ki = 405.8 nM T47768 C3H1NC 44434069 Ki = 91.49 nM T47768 C39AJW 44434071 Ki = 20.81 nM T47768 C38LOE 44434072 Ki = 11.86 nM T47768 CR9GY1 44434075 Ki = 12.03 nM T47768 CT6ZD0 44434077 Ki = 11.14 nM T47768 COI7A6 44434079 Ki = 7.55 nM T47768 C73FSU 44434081 Ki = 11.93 nM T47768 CKEY87 44434082 Ki = 18.33 nM T47768 CLZ68X 44434084 Ki = 42.03 nM T47768 CI2R7P 44434085 Ki = 24.42 nM T47768 C20PXC 44434087 Ki = 41.67 nM T47768 C1KB9R 44434088 Ki = 128.7 nM T47768 CLU1X5 44434089 Ki = 215.87 nM T47768 C72BXS 44434325 Ki = 0.62 nM T47768 C35HRS 44434326 Ki = 56.9 nM T47768 C0UK9Q 44434327 Ki = 4.23 nM T47768 C2CK7G 44434328 Ki = 15.4 nM T47768 C5J8VH 44434329 Ki = 8.88 nM T47768 C8CZX7 44434330 Ki = 76.5 nM T47768 C9DF1X 44434331 Ki = 129.1 nM T47768 C7CKX3 44434332 Ki = 1 nM T47768 CNFH86 44434333 Ki = 0.42 nM T47768 C5OW8M 44434334 Ki = 0.55 nM T47768 CS6BH9 44434335 Ki = 0.125 nM T47768 C61SUX 44434336 Ki = 0.66 nM T47768 CB2AQ4 44434932 Ki > 2500 nM T47768 C81KMS 44434933 Ki > 2500 nM T47768 COEG19 44434934 Ki = 1076.86 nM T47768 C9XW8Q 44434935 Ki > 2500 nM T47768 C4N9OY 44434936 Ki > 2500 nM T47768 C5UG8I 44434937 Ki > 2500 nM T47768 CGLY08 44434938 Ki = 20.55 nM T47768 C92WQA 44434939 Ki = 234.53 nM T47768 C04LKG 44434940 Ki = 52.29 nM T47768 CT95NA 44434941 Ki = 57.15 nM T47768 CGKC17 44434942 Ki = 52.27 nM T47768 CVF9O5 44434943 Ki = 389.49 nM T47768 CUA32P 44434944 Ki = 16.56 nM T47768 CRBX46 44434945 Ki = 18.47 nM T47768 CD0R6I 44434947 Ki > 1000 nM T47768 CIN4E6 44434948 Ki > 1000 nM T47768 CT30KJ 44437601 Ki = 57 nM T47768 C1EHS4 44437602 Ki = 60 nM T47768 CX5O0J 44437604 Ki = 9 nM T47768 CWOJ02 44437605 Ki = 113 nM T47768 CK73VO 44437606 Ki = 138 nM T47768 CJ1ST3 44437610 Ki = 54 nM T47768 CFH6A5 44437613 Ki = 188 nM T47768 C0M9SC 44437615 Ki = 271 nM T47768 CFN8Z9 44437617 Ki = 103 nM T47768 CTK2S0 44437619 Ki = 23 nM T47768 C4PK1O 44437623 Ki = 271 nM T47768 CP4HR6 44437626 Ki = 106 nM T47768 CA5S2P 44437627 Ki = 172 nM T47768 CKEG06 44437628 Ki = 122 nM T47768 CT7V0O 44437629 Ki = 1701 nM T47768 C45ZTN 44437630 Ki = 62 nM T47768 CQKL94 44437636 Ki = 125 nM T47768 C43URV 44437637 Ki = 70 nM T47768 CJ8L4A 44437638 Ki = 46 nM T47768 CNBQ93 44437639 Ki = 289 nM T47768 C2AV5I 44437640 Ki = 272 nM T47768 CN3R5G 44437641 Ki = 161 nM T47768 C6NA9R 44437642 Ki = 238 nM T47768 CH5RW4 44437643 Ki = 245 nM T47768 C7RIC8 44437644 Ki = 75 nM T47768 C5IL8O 44437645 Ki = 180 nM T47768 CX1S4V 44437646 Ki = 199 nM T47768 CV19NL 44437647 Ki = 432 nM T47768 C02YET 44437648 Ki = 100 nM T47768 CJ2PH5 44437649 Ki = 119 nM T47768 CVH1I9 44437652 Ki = 108 nM T47768 C0ME9B 44437654 Ki = 34 nM T47768 CRKH10 44437656 Ki = 16 nM T47768 CZB4Q9 44438912 Ki = 887 nM T47768 C7RD2E 44438916 Ki = 133 nM T47768 CNL30S 44438917 Ki = 37.4 nM T47768 C5D4NZ 44438920 Ki = 74 nM T47768 CA2LD5 44438921 Ki = 355 nM T47768 C6H7AD 44438922 Ki = 244 nM T47768 CRN3W4 44438961 Ki = 22 nM T47768 CGYD89 44438962 Ki = 30 nM T47768 CZ48KD 44438963 Ki = 475 nM T47768 C2EGK7 44438964 Ki = 818 nM T47768 COX57F 44438965 Ki = 778 nM T47768 C9S2HB 44438966 Ki = 1109 nM T47768 C1HF6E 44438967 Ki = 5081 nM T47768 C3L7SB 44438968 Ki = 346 nM T47768 CE63GK 44438971 Ki = 1616 nM T47768 C8TVI4 44438974 Ki = 567 nM T47768 CPHS56 44438975 Ki = 3187 nM T47768 CK3Z5G 44438978 Ki = 787 nM T47768 CPA4U5 44438983 Ki = 5.1 nM T47768 C2TKY5 44438988 Ki = 72.3 nM T47768 CL7WN5 44438993 Ki = 11.1 nM T47768 C0A2OM 44439000 Ki = 49.1 nM T47768 CMQA60 44439001 Ki = 59.1 nM T47768 CH57IQ 44439874 Ki > 10000 nM T47768 CNS7T5 44439878 Ki > 10000 nM T47768 CF86GQ 44443051 Ki = 474 nM T47768 CHEI51 44443452 Ki = 47 nM T47768 CY78KN 44443453 Ki = 71 nM T47768 CF1IC2 44443454 Ki = 66 nM T47768 CDJ8T5 44444601 Ki = 0.084 nM T47768 C9N8VT 44444603 Ki = 0.98 nM T47768 C57TLG 44444604 Ki = 1.3 nM T47768 CBR38Y 44444613 Ki = 2.5 nM T47768 C56QDE 44448327 Ki = 34 nM T47768 CPW3J0 44448489 Ki = 27 nM T47768 CN9X6W 44448522 Ki = 52 nM T47768 C6TEA5 44448524 Ki = 5.9 nM T47768 CET3O5 44448563 Ki = 25 nM T47768 CT39QP 44450085 IC50 = 1400 nM T47768 C1SQ7M 44450086 IC50 = 520 nM T47768 CJLI69 44450262 Ki = 2.1 nM T47768 C4NFQ9 44450499 Ki = 10 nM T47768 CL78ZG 44451517 Ki = 56.23 nM T47768 CG2WD7 44451518 Ki = 144.54 nM T47768 CBK6R5 44451542 Ki = 83.18 nM T47768 CC36BM 44451543 Ki = 104.71 nM T47768 CKB0F9 44451569 Ki = 100 nM T47768 C2EJP0 44451572 Ki = 42.66 nM T47768 CYQ53B 44451573 Ki = 524.81 nM T47768 CGJ3R8 44451592 Ki = 181.97 nM T47768 CAC1G4 44451593 Ki = 38.9 nM T47768 CV26FM 44451594 Ki = 52.48 nM T47768 CKRM60 44451595 Ki = 38.9 nM T47768 C4S0BF 44451619 Ki = 77.62 nM T47768 CAVN40 44451620 Ki = 1023.29 nM T47768 C2NCL3 44451621 Ki = 42.66 nM T47768 CHPO59 44451647 Ki = 100 nM T47768 C70TSK 44451648 Ki = 47.86 nM T47768 CZ1R2D 44451649 Ki = 36.31 nM T47768 CF4SX9 44451673 Ki = 204.17 nM T47768 C3O8ZP 44451696 Ki = 95.5 nM T47768 C7VLH3 44451724 Ki = 120.23 nM T47768 CYIP73 44451748 Ki = 38.9 nM T47768 C2IS4W 44451777 Ki = 123.03 nM T47768 CST06H 44451779 Ki = 223.87 nM T47768 C4C9TD 44451805 Ki = 120.23 nM T47768 C5RLP6 44451837 Ki = 213.8 nM T47768 CO01GQ 44451872 Ki = 75.86 nM T47768 C7KL9C 44451895 Ki = 47.86 nM T47768 C25JHV 44451918 Ki = 44.67 nM T47768 C5W9PF 44452254 Ki = 6320 nM T47768 CVI7M0 44452281 Ki = 7300 nM T47768 CWAN90 44452282 Ki = 5700 nM T47768 C8KXY7 44452306 Ki = 250 nM T47768 CK1F5Z 44453675 Ki = 11 nM T47768 CRM8K4 44453699 IC50 = 3.8 nM T47768 CUIC24 44453700 Ki = 4.7 nM T47768 C6QV3U 44453726 IC50 = 5.3 nM T47768 C5HM3F 44453728 Ki = 2 nM T47768 CDY56P 44453750 Ki = 2.7 nM T47768 CO56PJ 44453779 Ki = 1.9 nM T47768 CO2XU7 44453801 Ki = 2.9 nM T47768 COI2B9 44453822 Ki = 0.63 nM T47768 CR1S3K 44453824 IC50 = 6.8 nM T47768 C4ID6Y 44453825 IC50 = 36 nM T47768 CBUE46 44453848 IC50 = 63 nM T47768 CZ7X2D 44453849 Ki = 23 nM T47768 CTEK70 44453879 Ki = 32 nM T47768 CH1D0B 44453880 Ki = 28 nM T47768 CA05FK 44453881 IC50 = 16 nM T47768 CTO26R 44453900 IC50 = 14 nM T47768 CN7B2P 44453901 IC50 = 10 nM T47768 C1PQA7 44453924 IC50 = 5.5 nM T47768 C81IOK 44453925 IC50 = 28 nM T47768 CXC09Y 44454967 IC50 = 97 nM T47768 C75SEP 44454968 IC50 = 190 nM T47768 C5LN9M 44454971 IC50 = 130 nM T47768 CIH52C 44455025 IC50 = 7670 nM T47768 CI5T8S 44455135 IC50 = 2590 nM T47768 CGI6A7 44455136 IC50 > 10000 nM T47768 CM9OW7 44455170 IC50 = 84 nM T47768 C8E4AF 44455171 IC50 > 10000 nM T47768 CH4N8R 44455206 IC50 > 10000 nM T47768 CEZR53 44455270 IC50 > 10000 nM T47768 CVDA26 44455301 IC50 = 8000 nM T47768 C0UC6P 44455338 IC50 = 190 nM T47768 C7B1KA 44455368 EC50 = 24900 nM T47768 C89COF 44455373 IC50 > 10000 nM T47768 CRFJ58 44455391 IC50 > 10000 nM T47768 CZL97F 44455426 Ki > 10000 nM T47768 CMNX58 44455445 IC50 = 130 nM T47768 C12XGE 44456400 Ki > 10000 nM T47768 C9KU1O 44456785 Ki = 0.06 nM T47768 C6PEF7 44456833 Ki = 1.2 nM T47768 CQ0WM7 44469273 IC50 > 5000 nM T47768 C4DL5C 44469677 IC50 > 10000 nM T47768 C0N2XB 44474938 Ki = 201 nM T47768 CL5NO6 44541248 Ki = 0.97 nM T47768 C6K3GX 44541249 Ki = 1.31 nM T47768 CVX16Z 44541250 Ki = 1.46 nM T47768 C29MSC 44541387 Ki = 7.43 nM T47768 CI9O3F 44541388 Ki = 3.75 nM T47768 C6TW8L 44541389 Ki = 9.68 nM T47768 C6T1UX 44551464 Ki = 0.82 nM T47768 C4SVU2 44561370 IC50 = 3200 nM T47768 CRJM24 44561454 IC50 = 7400 nM T47768 CXJK43 44561493 IC50 = 4400 nM T47768 CQKE48 44564372 Ki = 2.02 nM T47768 CL80WF 44570025 Ki = 5.2 nM T47768 C5W8ZR 44570027 EC50 = 101 nM T47768 C8BSQ4 44570028 EC50 = 4.2 nM T47768 C9ERN6 44570030 Ki = 7.1 nM T47768 CP2M8D 44570031 Ki = 0.77 nM T47768 CN7UA9 44570032 Ki = 400 nM T47768 CPA48R 44570066 Ki = 1.6 nM T47768 C5RWA8 44570068 IC50 = 58 nM T47768 CGK40O 44570070 Ki = 0.15 nM T47768 C6C0XR 44570071 Ki = 4.5 nM T47768 CT10RB 44570072 Ki = 2.5 nM T47768 C8P3SX 44570073 Ki = 2.6 nM T47768 CB01RQ 44570075 Ki = 18 nM T47768 CPO2R3 44570675 Ki = 11 nM T47768 C67IZG 44574538 Ki = 42 nM T47768 C5Q4HZ 44574539 Ki = 708 nM T47768 C74LHO 44574585 Ki = 57 nM T47768 CPL5V1 44574586 Ki = 535 nM T47768 C7K4PC 44574587 Ki = 384 nM T47768 C1JPH8 44574588 Ki = 104 nM T47768 CNCS12 44574629 Ki = 781 nM T47768 CJXE09 44574630 Ki = 1553 nM T47768 C2FO5H 44574631 Ki = 622 nM T47768 C5YQ6B 44574632 Ki = 306 nM T47768 CD18EP 44574671 Ki = 3586 nM T47768 CDS1G8 44574672 EC50 = 545 nM T47768 C6ZMS9 44574705 Ki = 627 nM T47768 CXQM01 44574708 Ki = 123 nM T47768 CW1GU7 44574743 Ki = 576 nM T47768 CL6UI1 44574744 Ki = 458 nM T47768 CKO8N4 44574745 Ki = 27 nM T47768 CLVU91 44574789 Ki = 996 nM T47768 C5JZK9 44574790 Ki = 100 nM T47768 CVZ6K3 44574848 Ki = 55 nM T47768 CA78KV 44574850 Ki = 59 nM T47768 CPH7D4 44574890 Ki = 50 nM T47768 CQL2E4 44574891 Ki = 215 nM T47768 C9C3ZJ 44574892 Ki = 333 nM T47768 CLG57R 44574958 Ki = 887 nM T47768 CLMH36 44574962 Ki = 60 nM T47768 CAW3R4 44574963 Ki = 57 nM T47768 CAWB12 44575043 Ki = 474 nM T47768 CZO5J4 44575091 Ki = 7255 nM T47768 CI6Y7U 44575092 Ki = 738 nM T47768 C4ZCX6 44576628 IC50 = 25 nM T47768 C8HF3V 44577045 Ki = 3800 nM T47768 CRME18 44577046 Ki = 20 nM T47768 CI1L7Y 44577047 Ki = 630 nM T47768 CDPS18 44577048 Ki = 0.55 nM T47768 C8OU4Q 44577049 Ki = 88 nM T47768 CGMC75 44577468 Ki = 0.55 nM T47768 CZUW31 44577469 Ki = 890 nM T47768 CES86D 44577470 Ki = 6.9 nM T47768 CU6ZT4 44577524 Ki = 44 nM T47768 CXS42P 44577525 Ki = 28 nM T47768 CWIG26 44577526 Ki = 88 nM T47768 CTIH86 44577527 Ki = 32 nM T47768 C76AQL 44580898 Ki = 8.3 nM T47768 C3S2XF 44580899 Ki = 5.7 nM T47768 C6Q3NU 44580900 Ki = 29.4 nM T47768 CSH7E8 44580901 Ki = 24.1 nM T47768 C6XOD8 44580932 Ki = 0.0298 nM T47768 CRK51Y 44581834 Ki > 10000 nM T47768 CG1DL2 44582176 Ki = 2.02 nM T47768 C3YMV4 44582184 Ki = 1.59 nM T47768 CKFX03 44582185 Ki = 5.58 nM T47768 CK8G4D 44582186 Ki = 123.23 nM T47768 CIX09B 44582198 Ki = 68.4 nM T47768 CC06XI 44582199 Ki = 1.44 nM T47768 CEUS82 44582200 Ki = 2.69 nM T47768 C28VHY 44582218 Ki = 225.27 nM T47768 CRCH48 44582675 Ki > 10000 nM T47768 CEJ4R8 44582676 Ki > 10000 nM T47768 C5QB4K 44582678 Ki > 10000 nM T47768 C01RCI 44582705 Ki = 2009 nM T47768 CM21UD 44583389 Ki = 210 nM T47768 C6YOC5 44583390 Ki = 48 nM T47768 CX1L5P 44583391 Ki = 2200 nM T47768 C7PCJ1 44583392 Ki > 1000 nM T47768 CAHK35 44583425 Ki = 770 nM T47768 C7VWA3 44583426 Ki > 1000 nM T47768 CNG34J 44583429 Ki > 1000 nM T47768 CHZ46N 44583430 Ki > 1000 nM T47768 CASI92 44583431 Ki > 1000 nM T47768 CLAR69 44583432 Ki > 1000 nM T47768 CW32EA 44586706 Ki = 2.15 nM T47768 C54LFC 44586707 Ki = 2.92 nM T47768 CT2HF3 44586708 Ki = 3.02 nM T47768 CJFK08 44586709 Ki = 15.4 nM T47768 CL82BP 44586711 Ki = 115 nM T47768 CMZ3G4 44586712 Ki = 121 nM T47768 CSVR74 44586714 Ki = 151 nM T47768 C95DXO 44586715 Ki = 148 nM T47768 CJ1V8O 44586716 Ki = 266 nM T47768 CJOH07 44586888 Ki = 6.7 nM T47768 CJS8F2 44586890 Ki = 2.7 nM T47768 CP2N8S 44586914 Ki = 0.32 nM T47768 C7P0XN 44586916 Ki = 2.3 nM T47768 CV9H6N 44586918 Ki = 0.061 nM T47768 CP8EX5 44586920 Ki = 15 nM T47768 C1I0RO 44586943 Ki = 0.22 nM T47768 C5KN8O 44586945 Ki = 55 nM T47768 CZ9NA4 44586947 Ki = 18 nM T47768 CH97QC 44586949 Ki = 21 nM T47768 C8A9WK 44586979 Ki = 10 nM T47768 CZ28KA 44586981 Ki = 16 nM T47768 CYC3Z6 44586983 Ki = 3.9 nM T47768 C1HA0F 44588005 Ki > 8000 nM T47768 CS1G0I 44588006 Ki = 560 nM T47768 CT3C8S 44588007 Ki = 1220 nM T47768 CDMZ71 44588493 Ki > 10000 nM T47768 CVCW78 44588494 Ki = 352 nM T47768 CN7OR6 44588495 Ki = 3210 nM T47768 CZIM85 44588496 Ki = 49 nM T47768 C6EQ3R 44590514 IC50 = 69 nM T47768 CEXW79 44590551 EC50 = 2600 nM T47768 C5UIT4 44590552 IC50 = 4862 nM T47768 CP83ZW 44590553 IC50 = 126 nM T47768 C1AP0B 44590554 IC50 = 443 nM T47768 C4U3AE 44590580 IC50 = 211 nM T47768 CBS8P1 44590581 IC50 = 151 nM T47768 C41SFR 44590582 IC50 = 181 nM T47768 CD70YK 44590629 IC50 = 100 nM T47768 CY36KS 44590630 IC50 = 58 nM T47768 C60XNA 44590631 IC50 = 245 nM T47768 CJ3R7Q 44590632 IC50 = 351 nM T47768 CMH26K 44590677 IC50 = 1122 nM T47768 CN8S5P 44590678 IC50 = 4828 nM T47768 CIG43Y 44590679 IC50 = 2800 nM T47768 CX0RK9 44590708 IC50 = 772 nM T47768 CFLP28 44591164 Ki = 0.31 nM T47768 C8ZC6O 44591193 Ki = 0.77 nM T47768 CEA9O2 44591194 Ki = 60 nM T47768 CER74Z 44591195 Ki = 10 nM T47768 CIU9T1 44591196 Ki = 9.5 nM T47768 CO3P8X 44591197 Ki = 2.5 nM T47768 CN5ZF8 44591198 Ki = 1.4 nM T47768 CZJ16A 44591987 Ki = 3.8 nM T47768 C6A1PL 44592015 Ki = 0.072 nM T47768 CB3VG2 44592016 Ki = 1.3 nM T47768 CXL41O 44592053 Ki = 0.52 nM T47768 C3VSJ2 44592054 Ki = 37 nM T47768 CNI1E9 44592056 Ki = 2 nM T47768 CUW6Q3 44592086 Ki = 0.16 nM T47768 C8DS7Q 44592087 Ki = 2.5 nM T47768 CU5GE1 44592088 Ki = 0.3 nM T47768 C9GRS1 44592089 Ki = 1.2 nM T47768 CPX7G6 44592124 Ki = 46 nM T47768 CTYR04 44593576 Ki = 1487 nM T47768 C30YUJ 44593682 Ki = 0.081 nM T47768 CDPU87 44596170 Ki = 0.88 nM T47768 CYS09M 44597323 Ki = 3500 nM T47768 C2EC4H 44597424 Ki = 600 nM T47768 CJ69LZ 44597425 Ki = 1330 nM T47768 C90DGE 44597428 Ki = 48 nM T47768 C3ASC5 44597529 Ki = 9.3 nM T47768 C6XHL0 44597530 Ki = 80 nM T47768 CAOX39 44597597 Ki = 0.95 nM T47768 C2C9LF 44597714 Ki = 0.47 nM T47768 CEOB85 44597715 Ki = 2.9 nM T47768 C1R3QC 44597828 Ki = 1.7 nM T47768 CRS74M 44597830 Ki = 8.6 nM T47768 C39PTC 44597831 Ki = 0.46 nM T47768 C14EJV 44597940 Ki = 47 nM T47768 CV0GR9 44599826 Ki = 94 nM T47768 C84NFS 44599828 Ki = 10 nM T47768 CI6CW8 44599979 Ki = 193 nM T47768 CFY8I6 44599981 Ki = 70 nM T47768 C2XQN6 44599984 Ki = 198 nM T47768 C0G4ON 44600135 Ki = 433 nM T47768 C24QEG 44600140 Ki = 378 nM T47768 CQO2U6 44600308 Ki = 391 nM T47768 C3Q0ZL 44601476 IC50 > 32000 nM T47768 CVH94R 44608034 IC50 = 10300 nM T47768 CH68PJ 44620907 IC50 > 32000 nM T47768 CNR3K1 44626294 IC50 = 410 nM T47768 C5ABG6 44626295 IC50 > 10000 nM T47768 C3DCT2 44626536 Ki = 23 nM T47768 CUZY73 44626538 Ki = 24 nM T47768 CG8W0U 44626542 Ki = 360 nM T47768 CY6D4O 44626643 Ki = 110 nM T47768 CB9JD0 44626647 Ki = 290 nM T47768 C25QXW 44626747 Ki = 330 nM T47768 C2NC5S 44626748 Ki = 6.8 nM T47768 C6GB5A 44626749 Ki = 76 nM T47768 CCZ89E 44626842 Ki = 24 nM T47768 CKRL83 44627034 Ki = 160 nM T47768 CBNJ20 44627035 Ki = 64 nM T47768 CVD03Q 44627135 Ki = 74 nM T47768 C8XG3W 44627136 Ki = 35 nM T47768 C8PK2F 44627248 Ki = 17 nM T47768 C81KJQ 44627363 Ki = 36 nM T47768 CLUP27 44627365 Ki = 36 nM T47768 C8NJR1 44627679 Ki = 180 nM T47768 C7CJM9 44627680 Ki = 0.71 nM T47768 CM49FS 44627786 Ki = 5.4 nM T47768 C81LTN 44627787 Ki = 0.31 nM T47768 CPTL91 44627788 Ki = 2.5 nM T47768 CZ6VP4 44627789 Ki = 16 nM T47768 CQZ0W4 44627899 Ki = 0.026 nM T47768 C6AR0U 44627902 Ki = 0.61 nM T47768 CK0T4Y 44627998 Ki = 0.58 nM T47768 C79JNE 44627999 Ki = 1.1 nM T47768 CVI57S 44628102 Ki = 3.9 nM T47768 CS8X1U 44665679 IC50 = 30900 nM T47768 CR3PL6 44665680 IC50 > 32000 nM T47768 CT5CK8 44665687 IC50 > 32000 nM T47768 C3HXK5 45100475 IC50 = 10300 nM T47768 C45PUQ 45102745 Ki = 30 nM T47768 C4LOY2 45115589 IC50 = 1390 nM T47768 CU8I6T 45263517 Ki = 35 nM T47768 CY0GS5 45264200 Ki = 2800 nM T47768 CVDQ53 45265789 Ki = 361 nM T47768 CSWI21 45265820 IC50 = 2730 nM T47768 CA2O3N 45268153 Ki = 309 nM T47768 C8BPX4 45269032 Ki = 412 nM T47768 C40CHQ 45269407 Ki = 1.85 nM T47768 CT1U4X 45270231 Ki = 0.56 nM T47768 C7HF9D 45271055 Ki = 1.1 nM T47768 CU84PI 45271534 Ki = 325 nM T47768 C7ZWN3 45272750 Ki = 1.19 nM T47768 CIL49C 45482634 Ki = 0.18 nM T47768 CS2D7I 45482869 Ki = 728 nM T47768 CAP40I 45483185 Ki = 4162 nM T47768 CMN6O9 45483211 Ki = 1188 nM T47768 CFR5M7 45483251 Ki = 3750 nM T47768 CL7KU2 45483259 Ki = 1541 nM T47768 C8DOR2 45483260 Ki = 831 nM T47768 CFU8K5 45483286 Ki = 3809 nM T47768 C1X8JY 45483646 Ki = 5036 nM T47768 CGOZ34 45483648 Ki = 7104 nM T47768 CI8M5T 45483656 Ki = 4711 nM T47768 CE13WZ 45483658 Ki = 2879 nM T47768 CEZJ19 45483659 Ki = 486 nM T47768 C43JND 45483664 Ki = 75 nM T47768 C49WAV 45483668 Ki = 462 nM T47768 CVC0G3 45483672 Ki = 1017 nM T47768 C0J4CG 45483978 Ki = 0.43 nM T47768 CFY46C 45483979 Ki = 3.7 nM T47768 CC69WR 45483986 IC50 = 0.81 nM T47768 CLMP13 45483987 IC50 = 0.11 nM T47768 C3TJ9O 45483988 IC50 = 4.25 nM T47768 CPO50D 45483989 IC50 = 0.38 nM T47768 CQ5G8V 45483990 IC50 = 5.23 nM T47768 CKB8H3 45483991 IC50 = 29.8 nM T47768 CT0Y4W 45485562 IC50 > 10000 nM T47768 CE9D2C 45485563 IC50 = 4500 nM T47768 CSML06 45485564 IC50 > 10000 nM T47768 CQU3S9 45485604 IC50 > 10000 nM T47768 CG5QJ0 45485614 IC50 = 340 nM T47768 CE4ZG1 45485619 IC50 = 5100 nM T47768 CSK1X6 45485620 IC50 > 10000 nM T47768 CCY98N 45485624 IC50 > 10000 nM T47768 CREQ49 45485653 IC50 > 10000 nM T47768 CTQ1U3 45485675 IC50 > 10000 nM T47768 C89UEA 45485826 Ki = 87 nM T47768 C76IZT 45485837 Ki = 2106 nM T47768 C2DRY1 45485876 Ki = 1596 nM T47768 CBW8D7 45485877 Ki = 1963 nM T47768 C2OE9C 45485974 Ki = 2533 nM T47768 CBP10O 45485982 Ki = 1299 nM T47768 CS2IC5 45485986 Ki = 4445 nM T47768 CGB37Y 45486011 Ki = 162 nM T47768 C1TJC6 45486012 Ki = 1549 nM T47768 CHQI57 45486013 Ki = 772 nM T47768 C0KXD9 45486018 Ki = 205 nM T47768 CF46MY 45486027 Ki = 130 nM T47768 C9DVC1 45486028 Ki = 289 nM T47768 C3EV6H 45486032 Ki = 126 nM T47768 CV1N7L 45486033 Ki = 309 nM T47768 C9F4WP 45486035 Ki = 472 nM T47768 CC6DZ4 45486042 Ki = 177 nM T47768 CE1MR2 45486046 Ki = 127 nM T47768 CW7I8C 45486055 Ki = 88 nM T47768 C5JE6L 45486062 Ki = 648 nM T47768 CL2QF9 45486070 Ki = 115 nM T47768 CM39DL 45486096 Ki = 181 nM T47768 C60VCS 45486101 Ki = 62 nM T47768 CGY05X 45486102 Ki = 1251 nM T47768 C6YS7G 45486258 Ki = 36 nM T47768 CER4H7 45486486 Ki = 6543 nM T47768 C8CKM0 45487174 Ki = 0.3 nM T47768 CSC23N 45487200 Ki = 30 nM T47768 CFC45O 45487206 Ki = 24 nM T47768 C3QU2C 45487384 IC50 > 5000 nM T47768 CO7VJ6 46190938 Ki = 380 nM T47768 CO0Z6H 46190939 Ki > 890 nM T47768 CV89LB 46226159 Ki > 890 nM T47768 COZ08F 46226176 Ki > 890 nM T47768 CL10HJ 46226250 Ki = 110 nM T47768 C3YHF0 46227961 Ki = 0.34 nM T47768 C7LW1S 46227963 Ki = 0.47 nM T47768 C9L6WI 46227966 Ki = 1.09 nM T47768 C4FH3T 46229771 Ki = 0.9 nM T47768 C0ZOF5 46229772 Ki = 4 nM T47768 C6RK5N 46230439 Ki = 740 nM T47768 CSD7C9 46230440 Ki = 795 nM T47768 CK4TO1 46230441 Ki = 1630 nM T47768 C7L1QA 46230532 Ki = 670 nM T47768 C5UZ4O 46230533 Ki = 4670 nM T47768 C2QE0Y 46230534 Ki > 2700 nM T47768 CDF6P8 46230535 Ki = 354 nM T47768 CC85FR 46237455 Ki > 1000 nM T47768 CMJ0K7 46237580 Ki = 1150 nM T47768 C3R4KL 46237583 Ki > 1000 nM T47768 CC0K6V 46237584 Ki > 1000 nM T47768 CSH53K 46237585 Ki > 1000 nM T47768 CQ6K9E 46237703 Ki > 1000 nM T47768 C0G6MX 46237708 Ki = 470 nM T47768 CNC81F 46237832 Ki = 180 nM T47768 C97MLP 46237834 Ki = 140 nM T47768 C45EPA 46237835 Ki = 6120 nM T47768 CAY07H 46237836 Ki = 650 nM T47768 CCP98G 46237837 Ki > 1000 nM T47768 CWMO26 46632087 EC50 = 433 nM T47768 CF6ZY0 46632150 EC50 = 3424 nM T47768 CPNX59 46782151 Ki = 814 nM T47768 CK4D7I 46865103 Ki = 3200 nM T47768 C6EX2B 46865104 Ki = 13000 nM T47768 C8OK1P 46867404 EC50 = 120 nM T47768 C0J5XV 46867466 Ki = 41.1 nM T47768 C9NGO7 46869046 IC50 = 5400 nM T47768 CO5NQ3 46877612 Ki = 14.9 nM T47768 CF9G0A 46877633 Ki = 20.8 nM T47768 C5A7HD 46877642 Ki = 5.76 nM T47768 CVU37F 46877653 Ki = 0.45 nM T47768 CG19YU 46877660 Ki = 0.54 nM T47768 CWT3O2 46877673 Ki = 1.4 nM T47768 CY8TW9 46877674 Ki = 5.2 nM T47768 CC40AZ 46877676 Ki = 1.4 nM T47768 C1V9KZ 46877677 Ki = 0.19 nM T47768 CK7CY0 46878243 Ki = 0.34 nM T47768 CUMN01 46878245 Ki = 0.2 nM T47768 CJR0C1 46878247 Ki = 0.35 nM T47768 CS2V6N 46879477 Ki = 3.7 nM T47768 C6R8JO 46879478 Ki = 108 nM T47768 C9URN3 46879536 Ki = 21 nM T47768 C5PW9I 46879537 Ki = 5.2 nM T47768 CW2N7P 46879538 Ki = 12 nM T47768 CGJS91 46879539 Ki = 346 nM T47768 C08CHW 46879578 Ki = 27 nM T47768 CNF9D6 46879579 Ki = 1.1 nM T47768 C8UD2Z 46879580 Ki = 2.2 nM T47768 C9E8YP 46879581 Ki = 107 nM T47768 C9GB7O 46879627 Ki = 527 nM T47768 CU2F0K 46879629 Ki = 3177 nM T47768 CS7BP4 46879630 Ki = 113 nM T47768 C06NBW 46879667 Ki = 7.3 nM T47768 C0WY3K 46879668 Ki = 19 nM T47768 C5L7DB 46879669 Ki = 5.8 nM T47768 CSG31K 46879670 Ki = 14 nM T47768 C7P4UE 46879716 Ki = 268 nM T47768 C9NR8Q 46880030 Ki = 1794 nM T47768 C0O1PU 46880031 Ki = 608 nM T47768 CDY2L8 46880032 Ki = 11 nM T47768 CK01VS 46880033 Ki = 34 nM T47768 CFXU43 46880088 Ki = 350 nM T47768 CDM4C0 46880089 Ki = 282 nM T47768 CA8JU6 46880090 Ki = 77 nM T47768 C7LX9B 46880114 Ki = 47 nM T47768 C2VS0K 46880116 Ki = 127 nM T47768 CI5D6H 46880152 Ki = 1883 nM T47768 CR35XL 46880155 Ki = 2707 nM T47768 CI6ZA1 46880237 Ki = 67 nM T47768 CID57V 46880238 Ki = 138 nM T47768 CG6UO7 46880239 Ki = 120 nM T47768 C4LCV8 46880270 Ki = 45000 nM T47768 C8T5GF 46880271 Ki > 200000 nM T47768 CWK29B 46880272 Ki = 49000 nM T47768 C7HT9Q 46880391 Ki = 7.1 nM T47768 CARP46 46880392 Ki = 0.95 nM T47768 C12DCB 46880393 Ki = 1.2 nM T47768 C65ALC 46880394 Ki = 17 nM T47768 CKQ94Y 46880395 Ki = 12 nM T47768 C5HDU1 46880396 Ki = 3.2 nM T47768 C82AOZ 46880397 Ki = 4.8 nM T47768 CW3F8K 46880398 Ki = 2.4 nM T47768 CKJD61 46880399 Ki = 0.24 nM T47768 C1RZ7T 46880400 Ki = 7.3 nM T47768 CV7K6J 46880401 Ki = 7.4 nM T47768 C49NWA 46880452 Ki = 0.21 nM T47768 C7JK5C 46880453 Ki = 70 nM T47768 CE6Y5T 46880454 Ki = 6.5 nM T47768 CK8A1O 46880462 Ki > 10000 nM T47768 C9KDP4 46880463 Ki > 10000 nM T47768 CODR73 46880498 Ki > 10000 nM T47768 CHJ5Y6 46880566 Ki > 10000 nM T47768 CE9PG2 46880567 Ki > 10000 nM T47768 C01PGO 46880568 Ki > 10000 nM T47768 CS7L4X 46880569 Ki > 10000 nM T47768 C0PXY7 46880628 Ki > 10000 nM T47768 CD37LU 46880629 Ki > 10000 nM T47768 CUY89F 46880630 Ki > 10000 nM T47768 C4P6XS 46880631 Ki > 10000 nM T47768 CJ53KF 46880672 Ki > 10000 nM T47768 CYJC08 46880673 Ki > 10000 nM T47768 C1RI9O 46880674 Ki > 10000 nM T47768 C7JB8W 46906000 IC50 = 190 nM T47768 C5ZDY3 46915370 Ki = 8900 nM T47768 C0YJ1U 46928474 Ki = 57 nM T47768 CQ86RS 46928475 Ki = 4.7 nM T47768 C0HQ9F 46928476 Ki = 86 nM T47768 CI86QW 46928478 Ki = 3 nM T47768 CR3O7S 46928581 Ki = 110 nM T47768 CCSB86 46930969 IC50 = 580 nM T47768 CV16YQ 47023707 Ki = 1290 nM T47768 CABL63 49765080 IC50 = 1826 nM T47768 C2LZJ0 49783209 Ki > 10000 nM T47768 C57SMG 49783415 Ki > 10000 nM T47768 C0TG6I 49783419 Ki > 10000 nM T47768 CYP36E 49799951 Ki > 1000 nM T47768 CTR1Y2 49799964 EC50 = 7.3 nM T47768 CDS18H 49799966 Ki = 4.8 nM T47768 C4FA1V 49799967 Ki = 1.6 nM T47768 CEG52T 49799968 EC50 = 13.5 nM T47768 C2H8LY 49799969 EC50 = 0.66 nM T47768 C3T6NH 49843555 Ki = 201 nM T47768 CXW97O 49865703 IC50 = 18513 nM T47768 CRG60N 49865732 IC50 = 16334 nM T47768 CZY2T3 49865733 IC50 = 10681 nM T47768 CI2W0D 49865783 IC50 = 3941 nM T47768 CUK35O 49865784 IC50 = 3077 nM T47768 CL0DR3 49865859 IC50 = 17039 nM T47768 CE15WQ 49865860 IC50 > 30000 nM T47768 C9HEP1 49865919 IC50 = 8084 nM T47768 CL6ZG8 49865920 IC50 = 17039 nM T47768 CC6VB8 49865921 IC50 > 23040 nM T47768 CHYN61 49865922 IC50 > 26704 nM T47768 CP8VQ6 49865971 IC50 = 419 nM T47768 CAI09G 49865972 IC50 = 8188 nM T47768 CFT26X 49866025 IC50 = 22230 nM T47768 C2RY0J 50878551 Ki < 10000 nM T47768 C1W6TV 50898777 Ki > 10000 nM T47768 CXMZ73 50898778 Ki > 10000 nM T47768 CG4SX0 50942591 Ki > 10000 nM T47768 C9Y5CM 50964436 Ki = 8690 nM T47768 CU63SQ 50994498 Ki = 456 nM T47768 C5D0NY 51002736 Ki = 6 nM T47768 C3OQP7 51002739 Ki = 14 nM T47768 CBPQ82 51002822 Ki = 4 nM T47768 CCTI18 51002823 Ki = 3 nM T47768 CFGZ31 51002824 Ki = 11 nM T47768 CSW52C 51002825 Ki = 459 nM T47768 C8OFC7 51002870 Ki = 2 nM T47768 CG7US6 51002874 Ki = 26 nM T47768 C0B8ZH 51002978 Ki = 16 nM T47768 C7FI2R 51002981 Ki = 47 nM T47768 C7QA4S 51003039 Ki = 76 nM T47768 CGU3H2 51003042 Ki = 265 nM T47768 C08HUZ 51003216 EC50 = 4.24 nM T47768 CXW86B 51003218 EC50 = 0.69 nM T47768 CW5Q7V 51003448 Ki = 25.12 nM T47768 CGR98N 51003449 Ki = 1.585 nM T47768 C9WEO3 51003467 Ki = 2.5 nM T47768 CNV2Q4 51004758 IC50 = 695 nM T47768 C1SK7C 51009928 IC50 = 611 nM T47768 CM2K7S 51042171 Ki = 4500 nM T47768 CE4KP1 51050257 Ki > 10000 nM T47768 CQ6SR3 51353734 Ki = 1.1 nM T47768 CDQ3I6 51353736 Ki = 7.4 nM T47768 C4GH6F 51353738 Ki = 24 nM T47768 CZ1CL5 51353740 Ki = 76 nM T47768 C3W7AJ 51353742 Ki = 15 nM T47768 CK07VQ 51353744 Ki = 4 nM T47768 C9JAE4 51356293 Ki = 2.7 nM T47768 C7MNL4 51356294 Ki = 2.4 nM T47768 C3S0LD 51356295 Ki = 21 nM T47768 C6OY1E 51356296 Ki = 9.1 nM T47768 C54EPI 51356297 Ki = 10 nM T47768 CAU84H 51356590 Ki = 9.9 nM T47768 CZ1GB9 51356591 Ki = 130 nM T47768 CE16YQ 51356593 Ki = 180 nM T47768 CGF0L6 51356594 Ki = 610 nM T47768 CY5A7R 51357141 Ki = 1.8 nM T47768 CQ5Y6C 51357143 Ki = 17 nM T47768 CYB1A0 51357420 Ki = 10 nM T47768 C38DJS 52210045 Ki = 10200 nM T47768 C0TCI3 52915030 IC50 = 1900 nM T47768 CK6GN5 52915031 IC50 = 1160 nM T47768 CXF14W 52915032 IC50 = 1320 nM T47768 C27KOF 52915269 IC50 = 3345 nM T47768 CQ71YX 52915270 IC50 = 5114 nM T47768 CH56XF 52915389 IC50 = 4453 nM T47768 C02UBO 52915390 IC50 = 2593 nM T47768 CP2M6E 52915391 IC50 = 1977 nM T47768 CPA43I 52915392 IC50 = 4339 nM T47768 C5OA9H 52915393 IC50 = 2171 nM T47768 CA3P2C 52915514 IC50 = 2755 nM T47768 CK39TQ 52915515 IC50 = 1402 nM T47768 C98UZW 52915516 IC50 = 5333 nM T47768 CLAS61 52915517 IC50 = 4885 nM T47768 C7FDE9 52915518 IC50 = 5999 nM T47768 C9YOD2 52915634 IC50 = 9978 nM T47768 C1ZHF3 52915635 IC50 = 325 nM T47768 CZB67C 52915636 IC50 = 7071 nM T47768 CE3IS2 52915637 IC50 = 1401 nM T47768 CYB6J8 52916598 IC50 = 468 nM T47768 CG1F9W 52916599 IC50 = 1590 nM T47768 C7NO2D 52916712 IC50 = 2505 nM T47768 CZ3K9S 52916713 IC50 = 1390 nM T47768 CI32WO 52916714 IC50 = 1038 nM T47768 C2VN8I 52937468 Ki = 0.15 nM T47768 C1M3SD 52941462 IC50 = 424 nM T47768 C58ART 52941549 IC50 = 9410 nM T47768 CYLC29 52942529 IC50 = 1046 nM T47768 CPOQ82 52942580 IC50 = 19001 nM T47768 C3YF5D 52942581 IC50 > 30000 nM T47768 CKN2U6 52942810 IC50 > 30000 nM T47768 C5V4DW 52943162 IC50 = 482 nM T47768 CNK14O 52943803 IC50 = 307 nM T47768 CRH1Q5 52943993 IC50 > 30000 nM T47768 CBW0A9 52944041 IC50 > 30000 nM T47768 C89GIK 52944552 IC50 = 2894 nM T47768 CP5A3T 52944907 IC50 > 24383 nM T47768 C54ZBG 52944974 IC50 = 1896 nM T47768 CV48KS 52945118 IC50 = 253 nM T47768 C1G0IP 52945138 IC50 = 19837 nM T47768 CWA1T5 52945160 IC50 = 4.8 nM T47768 CSZ4R3 52945588 IC50 = 659 nM T47768 CNGU78 52945626 IC50 = 2648 nM T47768 CG8CN4 52946340 IC50 = 21090 nM T47768 CFN7I8 52947509 IC50 = 1944 nM T47768 C41AYU 52947523 IC50 = 9432 nM T47768 CY06OH 52947573 IC50 = 8504 nM T47768 CY72CQ 52947593 IC50 = 16785 nM T47768 CFI96N 52947735 IC50 = 17554 nM T47768 CI63UL 52948240 IC50 = 7854 nM T47768 CAID24 52948615 IC50 > 30000 nM T47768 C15KNW 52948655 IC50 = 22931 nM T47768 C48RBH 52948719 IC50 = 9359 nM T47768 CZX5B9 52948735 IC50 = 576 nM T47768 CPN4Z8 52948969 IC50 = 2698 nM T47768 CVWY23 52949439 IC50 = 10854 nM T47768 C9V6GB 52950007 IC50 = 22696 nM T47768 C01KMG 52952006 Ki > 3200 nM T47768 CL1QG4 52952007 Ki > 4800 nM T47768 CET8Q0 52952008 Ki > 2500 nM T47768 C6X7WL 52952107 Ki > 2700 nM T47768 C4N9HF 52952108 Ki > 1700 nM T47768 CWC1N8 52952109 Ki > 3000 nM T47768 C7JB4Q 52952110 Ki > 3000 nM T47768 C2GPE5 52952207 Ki > 3000 nM T47768 C6NP1V 53233475 EC50 = 0.1 nM T47768 CMJ62D 53245590 Ki = 1540 nM T47768 CTU43X 53316968 Ki > 450 nM T47768 CCOD69 53316969 Ki = 16 nM T47768 CE3P7Y 53317205 Ki = 31.62 nM T47768 C0NKY7 53317262 Ki = 50.12 nM T47768 C7H8QK 53318490 Ki = 1995.26 nM T47768 C31ZOA 53318757 Ki = 100 nM T47768 CI6CQ0 53319615 Ki = 178 nM T47768 C6SY4G 53319616 Ki > 450 nM T47768 C3PW1V 53319617 Ki > 450 nM T47768 CB10OV 53319822 Ki = 5.012 nM T47768 CT8R3I 53319870 Ki = 25.12 nM T47768 C4XD5Q 53319871 Ki = 12.59 nM T47768 CK73JR 53320122 Ki = 1.75 nM T47768 CY5MG9 53321111 Ki = 630.96 nM T47768 CD14AE 53321176 Ki = 398.11 nM T47768 C6X9OT 53321653 Ki > 3981.07 nM T47768 C2EV1S 53322245 Ki > 450 nM T47768 C1L8IV 53322246 Ki > 450 nM T47768 CRN26Z 53322438 Ki = 39.81 nM T47768 CZY2G3 53322439 Ki = 25.12 nM T47768 CMOL62 53322496 Ki = 15.85 nM T47768 CLDI90 53323074 Ki = 1.1 nM T47768 C30TBO 53323800 Ki = 50.12 nM T47768 CS9I6Z 53323801 Ki = 100 nM T47768 CGI94L 53323802 Ki = 12.59 nM T47768 C5I4KQ 53323803 Ki = 125.89 nM T47768 C0ZJ1T 53323804 Ki = 7.943 nM T47768 CV5EC1 53323805 Ki = 7.943 nM T47768 C7Z4KR 53323841 Ki > 3162.28 nM T47768 C32YWL 53324045 Ki = 70 nM T47768 C0MD2H 53324890 Ki = 302 nM T47768 CJ59GU 53325079 Ki = 10 nM T47768 CH37ZT 53325227 Ki > 10000 nM T47768 CRQF15 53325242 Ki = 356 nM T47768 C5E7LW 53325608 Ki = 229 nM T47768 CL5WG8 53325725 Ki = 3.5 nM T47768 CRZ76L 53326167 Ki = 128 nM T47768 CLP1Q0 53326367 Ki = 79.43 nM T47768 C7ETI8 53326368 Ki = 50.12 nM T47768 CI3K7N 53326835 Ki = 50.12 nM T47768 CA3KL4 53388149 Ki = 0.58 nM T47768 C0TIQ5 53388316 Ki = 0.73 nM T47768 CFE6S4 53465409 Ki = 1260 nM T47768 CT62EG 53465411 Ki = 751 nM T47768 CU04GB 53465412 Ki = 684 nM T47768 C7V4ME 53465413 Ki = 1007 nM T47768 C89NMJ 53465486 Ki = 740 nM T47768 CDV57J 53465487 Ki = 89 nM T47768 CN2P0M 53465488 Ki = 101 nM T47768 C03LXZ 53465489 Ki > 3000 nM T47768 C7JV2P 53465490 Ki = 66 nM T47768 C0NW4J 53465491 Ki = 207 nM T47768 C6C1FN 53465556 Ki = 32 nM T47768 CQ5F0H 53465557 Ki = 932 nM T47768 CW8XR1 53465558 Ki > 3000 nM T47768 CL27OF 53465559 Ki = 112 nM T47768 CB7F1V 53465560 Ki = 763 nM T47768 CF87WN 53465561 Ki > 3000 nM T47768 CJX6G9 53465633 Ki > 1000 nM T47768 C5W8PL 53465634 Ki > 3000 nM T47768 CR8FE6 53465635 Ki > 3000 nM T47768 CBFI98 53465636 Ki = 1327 nM T47768 C6MS1K 53465637 Ki > 3000 nM T47768 CUR52F 53465638 Ki = 163 nM T47768 CI18GY 53465639 Ki = 735 nM T47768 C8D7CS 53465710 Ki = 39 nM T47768 CR1VM6 53466534 Ki = 508 nM T47768 CMOZ61 53475319 Ki = 745 nM T47768 CO8ZP9 53498895 Ki = 5700 nM T47768 CE36IO 53521863 EC50 = 200 nM T47768 C70BZV 54580938 Ki = 0.089 nM T47768 CYEC84 54581367 Ki = 2700 nM T47768 C3I0HF 54582933 Ki = 0.82 nM T47768 C9G8RT 54582934 Ki = 8.8 nM T47768 CX0O1G 54583374 Ki = 1.1 nM T47768 C7L9JS 54583594 Ki = 18 nM T47768 CHA7T8 54584041 Ki = 0.15 nM T47768 C96ISF 54584882 Ki = 0.14 nM T47768 CKUH91 54585844 Ki = 0.55 nM T47768 C6MHV9 54585845 Ki = 2.5 nM T47768 CV86NQ 54586810 Ki = 0.26 nM T47768 CQ83TL 54596311 Ki = 0.36 nM T47768 C3EP9X 54669894 EC50 = 0.00174 nM T47768 C50VRZ 54678117 Ki = 3.4 nM T47768 C0IT4S 54678127 Ki = 4 nM T47768 CQIS61 54678129 Ki = 1.1 nM T47768 CH1LY5 54678130 Ki = 1 nM T47768 CGVW28 54718272 Ki = 5.1 nM T47768 CXF1G9 54751920 Ki = 5.9 nM T47768 CNT03F 54754507 Ki = 3.6 nM T47768 CROS84 54756989 EC50 = 2.6 nM T47768 C2ISE6 54756990 Ki = 2.19 nM T47768 C7F6EC 54757387 EC50 = 0.0832 nM T47768 C6EN8F 55433787 EC50 = 110 nM T47768 CQU87I 56589659 EC50 = 1.8 nM T47768 CHZ1D7 56589680 EC50 = 113 nM T47768 C28AED 56655502 Ki = 35.8 nM T47768 CCN2E8 56658044 EC50 = 6.1 nM T47768 CJW5C1 56658452 Ki = 0.67 nM T47768 CP37LM 56659141 Ki = 109 nM T47768 C69VIF 56661555 Ki = 13.2 nM T47768 CJ2MA7 56663008 Ki = 0.7 nM T47768 CUE0R7 56664847 IC50 = 8.2 nM T47768 CDKP63 56664973 Ki = 2.14 nM T47768 CEW3K4 56665405 Ki = 0.57 nM T47768 CR64WX 56665407 Ki = 0.85 nM T47768 C3QLV1 56666529 Ki = 384 nM T47768 C4QM3N 56668405 Ki = 14.3 nM T47768 C8O7MT 56668839 Ki = 0.1 nM T47768 CL21RS 56669900 Ki = 1.75 nM T47768 CO18SG 56669938 Ki > 2800 nM T47768 COEA65 56670013 Ki = 168 nM T47768 C9SY1A 56672310 Ki = 0.39 nM T47768 C2NQJ4 56673010 Ki = 1.69 nM T47768 CA4VH9 56673522 Ki = 3.5 nM T47768 CD9JK4 56675713 Ki = 0.45 nM T47768 CG1XO8 56676328 Ki = 21 nM T47768 C45KMW 56676759 Ki > 2800 nM T47768 C0WVZ6 56676760 Ki = 167 nM T47768 CVXJ29 56676761 Ki = 486 nM T47768 C7EFI9 56678759 IC50 = 11 nM T47768 CS8Z1G 56678760 IC50 = 20.8 nM T47768 CQZ75Y 56678873 Ki = 67 nM T47768 CZ6B0O 56678874 Ki = 1.1 nM T47768 C15FOK 56679008 Ki = 0.63 nM T47768 CDG30L 56680069 Ki = 250 nM T47768 CX8F2N 56681954 Ki = 5.56 nM T47768 C2A4MQ 56681955 Ki = 10.5 nM T47768 CK52GV 56682330 Ki = 0.87 nM T47768 C95LAM 56834761 EC50 = 0.079 nM T47768 CRX31L 56840667 Ki = 481 nM T47768 CQ2O4U 56849549 Ki = 52.7 nM T47768 CCMS01 56849550 Ki = 43.1 nM T47768 C7VT5K 56849551 Ki = 107 nM T47768 C2Y9CE 56851423 Ki = 232 nM T47768 C34PMD 56851424 Ki = 39.6 nM T47768 CN32ZB 56851582 Ki = 31.5 nM T47768 CY9DH2 56851583 Ki = 25.8 nM T47768 CC3JS8 56851584 Ki > 500 nM T47768 C9E6CU 56851585 Ki > 500 nM T47768 C1ZOM5 56851586 Ki = 101 nM T47768 CL45WN 57345320 IC50 = 14900 nM T47768 C5JKZ3 57345673 Ki = 0.08 nM T47768 CS1K0A 57391716 Ki = 4.6 nM T47768 CZ1EH9 57391826 IC50 > 10000 nM T47768 CHSW27 57392492 IC50 = 2330 nM T47768 CX89LJ 57392493 IC50 = 1200 nM T47768 CJ38ZY 57393448 Ki = 315 nM T47768 C6D7UA 57394195 IC50 = 1250 nM T47768 C3K5FX 57394196 IC50 = 6800 nM T47768 C4QZH8 57394197 IC50 = 140 nM T47768 CS02AB 57395174 Ki = 138 nM T47768 CSE78X 57395267 IC50 = 480 nM T47768 C4NI1O 57395962 IC50 = 180 nM T47768 C3BR0J 57396943 Ki = 346 nM T47768 C12ASH 57396944 Ki = 22 nM T47768 CNX73U 57397760 IC50 = 33 nM T47768 CC8EV2 57397761 IC50 = 490 nM T47768 C1HF3V 57397762 IC50 = 340 nM T47768 C84EKV 57398678 IC50 = 420 nM T47768 CP8KQ7 57399426 IC50 = 990 nM T47768 C4H6LZ 57399427 IC50 = 1600 nM T47768 CLNB91 57399428 IC50 = 330 nM T47768 C7T9ID 57399429 IC50 = 350 nM T47768 C0I4SM 57400106 Ki = 0.3 nM T47768 C95NKZ 57400481 IC50 = 200 nM T47768 CMP1F7 57400482 IC50 = 220 nM T47768 C3QF9I 57401062 Ki = 0.56 nM T47768 CVXU49 57401184 IC50 = 63 nM T47768 CR3K6X 57401866 Ki = 2.5 nM T47768 C8RX7I 57402172 Ki = 74 nM T47768 C5X0LN 57402288 IC50 > 8300 nM T47768 CUL3W2 57402462 Ki = 605 nM T47768 CT1IN3 57412337 Ki = 9.5 nM T47768 C7F4PN 57412339 Ki = 26 nM T47768 CTO37U 57412341 Ki = 17 nM T47768 C0UZ3G 57412343 Ki = 3.2 nM T47768 C3JL0D 57412421 Ki = 45 nM T47768 C10ZIE 57412591 Ki = 13 nM T47768 C8A1JR 57412593 Ki = 8.5 nM T47768 C5Q7KD 57412595 Ki = 7 nM T47768 CU80IK 57412597 Ki = 60 nM T47768 C2WG9D 57412599 Ki = 44 nM T47768 C5D6QU 57412771 Ki = 150 nM T47768 CNI7Y9 57412772 Ki = 2.7 nM T47768 C21LRT 57412773 Ki = 0.69 nM T47768 CFB58K 57412848 Ki = 0.86 nM T47768 CTV4X5 57412849 Ki = 1.7 nM T47768 CSYI37 57412850 Ki = 0.34 nM T47768 CJI87G 57412851 Ki = 1.2 nM T47768 CCB0G9 57412852 Ki = 0.51 nM T47768 CDV4H9 57412853 Ki = 0.17 nM T47768 CAO20P 57412942 Ki = 0.43 nM T47768 CF1LC3 57412943 Ki = 1.7 nM T47768 CYN92K 57412944 Ki = 0.32 nM T47768 C54XQG 57412945 Ki = 0.35 nM T47768 C0GL5A 57412946 Ki = 1.9 nM T47768 CGN29J 57413036 Ki = 0.16 nM T47768 C5ZHT6 57413037 Ki = 0.28 nM T47768 CP9L1N 57413038 Ki = 0.42 nM T47768 CP6G5F 57413039 Ki = 14 nM T47768 CH0B1F 57413040 Ki = 13 nM T47768 CQW92S 57822038 Ki = 1.6 nM T47768 C8XF6W 57822045 Ki = 7.3 nM T47768 CV1Y9U 57822053 Ki = 46.1 nM T47768 CTE6B5 57822082 Ki = 9.8 nM T47768 CELJ49 57822098 Ki = 93.6 nM T47768 C60ZHX 57822157 Ki = 16.5 nM T47768 CK0P5N 57822243 Ki = 19.4 nM T47768 C0J3LY 57900041 Ki = 0.064 nM T47768 C6AWU4 57900045 Ki = 0.82 nM T47768 C7MI3X 58046500 Ki = 9800 nM T47768 CFXC84 58046524 Ki = 1490 nM T47768 CI5H3N 58268566 Ki > 375 nM T47768 C6Z9JF 58268629 Ki > 400 nM T47768 C7EFU5 58443192 Ki = 0.23 nM T47768 C73BYR 58443217 Ki = 0.059 nM T47768 C5V8NC 58443218 Ki = 0.23 nM T47768 C7Z8SF 58443225 Ki = 0.0056 nM T47768 CS70GT 58443229 Ki = 0.64 nM T47768 CFXB82 58443230 Ki = 0.43 nM T47768 C4FKN0 58443234 Ki = 0.0016 nM T47768 CW81HV 58443235 Ki = 0.12 nM T47768 C2PJ4N 59271992 IC50 = 1000 nM T47768 CUE79I 59272004 IC50 > 2000 nM T47768 CJO8H7 59345567 EC50 = 61 nM T47768 C6GA5O 60150457 Ki > 10000 nM T47768 C7N0KO 60150458 Ki > 1000 nM T47768 C6G5TY 60154189 Ki > 400 nM T47768 C8MS6N 60154191 Ki > 400 nM T47768 CW63KM 60154192 Ki > 400 nM T47768 C2QX6R 60154193 Ki > 400 nM T47768 CD46EJ 60154264 Ki > 400 nM T47768 CEB0P5 60166738 Ki = 14.9 nM T47768 CYUB94 60168107 EC50 = 0.0334 nM T47768 CMAP25 60170608 EC50 = 36.5 nM T47768 C9AB5E 60170609 EC50 = 0.16 nM T47768 CQ3I4L 60170610 Ki = 15.7 nM T47768 C9VYO5 60170611 EC50 = 7.35 nM T47768 CU35KA 60170688 Ki = 7.12 nM T47768 CF8M6H 60170689 EC50 = 0.72 nM T47768 C2JUE9 60170691 Ki = 4.83 nM T47768 C8U1DO 60170774 Ki = 7.73 nM T47768 CW4P3F 60170775 EC50 = 0.0342 nM T47768 CR1GS9 60170776 Ki = 26 nM T47768 CY7E9U 60170777 Ki = 27.4 nM T47768 CVPG71 60561198 EC50 = 16 nM T47768 C0L5HT 62706594 Ki = 5.41 nM T47768 CJHB32 62706595 Ki = 110 nM T47768 C9EIX4 62706596 Ki = 170 nM T47768 C04WBM 62706597 Ki = 2900 nM T47768 CS9KV1 62706598 Ki = 27 nM T47768 CX72ZW 62706764 Ki = 12 nM T47768 C24YCI 62706765 Ki = 42 nM T47768 CEL48Q 62706766 Ki = 48 nM T47768 C7XEA4 62706767 Ki = 7.5 nM T47768 CC5B6H 62706768 Ki = 7.8 nM T47768 C98XRD 66911347 Ki = 44.5 nM T47768 CZ63PG 66986460 Ki = 3.1 nM T47768 CR50DU 67157108 Ki = 0.1585 nM T47768 C87KCO 67182916 Ki = 0.1259 nM T47768 C19UXP 67183276 Ki = 0.1 nM T47768 C1TEC7 67183439 Ki = 0.1995 nM T47768 CF6RB3 67183527 Ki = 0.1995 nM T47768 C5EV8P 67183538 Ki = 0.1 nM T47768 CNJ41I 67183562 Ki = 0.631 nM T47768 CY9R3L 67183680 Ki = 0.1 nM T47768 CYT8L5 67184545 Ki = 0.7943 nM T47768 CM3JW0 67184580 Ki = 0.2512 nM T47768 CYA6S5 67184933 Ki = 1.585 nM T47768 C7KLB6 68196155 EC50 = 2.7 nM T47768 C9YUL1 68314000 EC50 = 630.96 nM T47768 CL1M4R 68314236 EC50 = 199.53 nM T47768 C32BZW 68314305 EC50 = 31.62 nM T47768 C0SV2K 68314306 EC50 = 501.19 nM T47768 CI64QT 68314329 EC50 = 1584.89 nM T47768 C8KI5V 68314366 EC50 = 1258.93 nM T47768 CWD91X 68314457 EC50 = 158.49 nM T47768 CM46VH 68314562 EC50 = 158.49 nM T47768 CYBC09 68775633 Ki = 2460 nM T47768 CCK5Z9 68776073 Ki = 2800 nM T47768 CHF83Z 68776748 Ki = 2800 nM T47768 CJAH92 68777672 Ki = 5100 nM T47768 CA56LT 68777734 Ki = 3335 nM T47768 CKX63G 68777945 Ki = 2200 nM T47768 CVF8G6 68778394 Ki = 4690 nM T47768 C1I8MB 68778890 Ki = 740 nM T47768 C27KQI 68779363 Ki = 2260 nM T47768 C83YWM 68779815 Ki = 2300 nM T47768 CK4MH1 68782313 Ki = 1300 nM T47768 C89TSB 68867300 Ki = 4.34 nM T47768 CF5I0R 68917692 Ki = 1.95 nM T47768 C4DO7H 70158365 Ki > 890 nM T47768 C30HMT 70681352 Ki > 10000 nM T47768 CS1E7F 70681353 Ki = 3400 nM T47768 CPE62M 70682348 Ki > 450 nM T47768 C58AOU 70682351 Ki = 238 nM T47768 C9AW5C 70682920 Ki > 100 nM T47768 C5JLS9 70683421 Ki = 2600 nM T47768 CJ79UV 70683422 Ki > 10000 nM T47768 CH64DO 70683436 Ki > 1000 nM T47768 CZW6K5 70683437 Ki > 10000 nM T47768 CX3M0F 70683438 Ki > 1700 nM T47768 C6G0SO 70684433 Ki = 318 nM T47768 CLY56A 70684435 Ki > 450 nM T47768 C8U1PW 70684436 Ki = 80.7 nM T47768 CXY52W 70685543 Ki > 1000 nM T47768 C60FVD 70685544 Ki = 2530 nM T47768 CU7V8F 70685545 Ki > 10000 nM T47768 CWAL85 70686573 Ki = 397 nM T47768 CQL0S6 70687673 Ki > 10000 nM T47768 CY8DQ1 70687674 Ki > 10000 nM T47768 CE6K8V 70687698 Ki = 3600 nM T47768 CI61FE 70688692 Ki = 235 nM T47768 C08OUK 70688693 Ki > 450 nM T47768 C3HAX5 70688697 Ki = 139 nM T47768 CS86LY 70689742 Ki > 1000 nM T47768 CF7PZ4 70690755 Ki = 138 nM T47768 CMNL89 70690756 Ki = 29.8 nM T47768 CWB17N 70690757 Ki = 502 nM T47768 CTB4I1 70690760 Ki = 82.1 nM T47768 CY6E2Q 70691339 IC50 = 3920 nM T47768 CCQ5Z6 70691889 Ki = 4800 nM T47768 C3E4FO 70692893 Ki > 450 nM T47768 C1A7LO 70693567 EC50 = 1.9 nM T47768 C9PQ4F 70693930 Ki > 10000 nM T47768 CU60IL 70694933 Ki > 450 nM T47768 CWO5F0 70695375 Ki > 400 nM T47768 CRG52J 70695535 Ki > 10000 nM T47768 C2V8UI 70696034 Ki = 3090 nM T47768 CJ07AO 70696988 Ki > 450 nM T47768 CV0P1X 70696991 Ki = 67.2 nM T47768 CFQ8Y9 70696992 Ki = 28.4 nM T47768 CG3U7F 70697391 Ki > 400 nM T47768 CJ5DI4 70822235 Ki = 23.03 nM T47768 CI8M5U 70834572 Ki > 10000 nM T47768 CEOQ43 71229805 Ki = 0.71 nM T47768 CIK86Q 71230334 Ki = 1.3 nM T47768 CLA6O8 71449105 IC50 = 1010 nM T47768 C2TY6U 71449133 Ki = 0.14 nM T47768 CEB0P4 71449173 IC50 = 635 nM T47768 C8HV9A 71449570 Ki = 400 nM T47768 C3GCX4 71449910 Ki = 760 nM T47768 CYG07C 71449995 Ki = 1.25 nM T47768 CK69PO 71450043 Ki = 2.13 nM T47768 C4TVF1 71450063 Ki > 100000 nM T47768 CHQZ46 71450134 Ki = 13 nM T47768 CSC3R7 71450213 Ki = 412 nM T47768 C6DU5P 71450548 Ki = 2330 nM T47768 C9VZ8J 71450550 Ki = 5325 nM T47768 CJL59V 71450766 Ki = 0.064 nM T47768 C4BP5T 71450767 Ki = 0.18 nM T47768 C6JMZ4 71450851 Ki = 229 nM T47768 CQ6M2A 71450900 IC50 = 1050 nM T47768 C6ZX3S 71450925 Ki = 1.69 nM T47768 C5YIC1 71450926 Ki = 2.96 nM T47768 C2R7GS 71450927 Ki = 0.68 nM T47768 CMB7X9 71450932 Ki = 37.2 nM T47768 CNP02X 71450939 Ki = 0.67 nM T47768 C7FKC6 71451409 Ki = 1.6 nM T47768 C3GX1O 71451410 Ki = 3.87 nM T47768 C08KHB 71452040 Ki = 826 nM T47768 C0XW8E 71452041 Ki = 542 nM T47768 CDTW09 71452387 Ki = 4780 nM T47768 CYU3K7 71452742 Ki = 0.43 nM T47768 C4B6HU 71452746 Ki = 76.3 nM T47768 CYFH30 71452786 IC50 = 587 nM T47768 C2YWE8 71453373 EC50 = 0.84 nM T47768 CQY10P 71453677 Ki = 0.43 nM T47768 CRY4A1 71453704 Ki > 100000 nM T47768 CYOS40 71453706 Ki > 100000 nM T47768 CW0H5Q 71453774 Ki = 84 nM T47768 CZ08WY 71454361 Ki = 0.0049 nM T47768 CG82PA 71454362 Ki = 0.0071 nM T47768 CM0H5E 71454460 Ki = 115 nM T47768 CXQ1G0 71454513 Ki = 0.74 nM T47768 CGM86O 71454514 Ki = 0.19 nM T47768 CQ5JE8 71454515 Ki = 11.3 nM T47768 CI16ON 71454516 Ki = 34.2 nM T47768 CO01LV 71454517 Ki = 0.22 nM T47768 C09IMN 71454521 Ki > 1900 nM T47768 CCKA54 71454553 IC50 = 1140 nM T47768 CYJ9X8 71454554 IC50 = 1240 nM T47768 CI0G3P 71455268 Ki > 10000 nM T47768 C6F9KY 71455270 Ki > 10000 nM T47768 CN3EX8 71455429 Ki > 100000 nM T47768 CW63BC 71455505 Ki = 3.03 nM T47768 C89UMR 71455506 Ki = 0.41 nM T47768 C9WB3S 71455767 EC50 = 6 nM T47768 C6G2HC 71455894 Ki = 1269 nM T47768 CFBC49 71455896 Ki = 3415 nM T47768 C83WJY 71456105 Ki = 1.8 nM T47768 CQ0UG3 71456106 Ki = 0.0056 nM T47768 CF9HA1 71456174 Ki = 1.5 nM T47768 C42HSQ 71456256 Ki = 33.4 nM T47768 C8FXZ5 71456257 Ki = 10.2 nM T47768 CDQM86 71456258 Ki = 51.1 nM T47768 CXZ2V8 71456262 EC50 = 0.04 nM T47768 C1G7OM 71456308 IC50 = 8240 nM T47768 C2X3AN 71456309 IC50 = 8130 nM T47768 C5E1ST 71457059 Ki = 1010 nM T47768 C42MER 71457207 Ki = 74000 nM T47768 C3XIP8 71457209 Ki > 100000 nM T47768 C9UVJ1 71457210 Ki = 5.6 nM T47768 CLN75C 71457288 Ki = 41.9 nM T47768 CH4Y5I 71457289 Ki = 7.89 nM T47768 CPUO14 71457290 Ki = 1.04 nM T47768 C4KD6E 71457291 Ki = 2.58 nM T47768 C0R8UO 71457292 Ki = 0.94 nM T47768 CDSX56 71457372 Ki = 788 nM T47768 CP7JI0 71457691 Ki = 7474 nM T47768 C9GQO5 71458037 IC50 = 1150 nM T47768 CSJ4A1 71458063 Ki = 0.23 nM T47768 CG98LJ 71458064 Ki = 0.48 nM T47768 CV74RO 71458065 EC50 = 5.2 nM T47768 CP6DQ7 71458116 IC50 = 2870 nM T47768 C92YCB 71458142 IC50 = 1940 nM T47768 CQ46CG 71458581 Ki = 0.73 nM T47768 C8LNZ6 71459067 Ki > 100000 nM T47768 CK5T4P 71459604 Ki = 5392 nM T47768 C7X9YH 71459820 Ki = 0.3 nM T47768 CA1N5D 71459821 Ki = 0.021 nM T47768 CNCA72 71459902 Ki = 571 nM T47768 CQ52LR 71459947 Ki = 0.63 nM T47768 CFR1T9 71459948 Ki = 2.61 nM T47768 CUID52 71459949 Ki = 1.98 nM T47768 C0TP7N 71459950 Ki = 12.8 nM T47768 CHS4D2 71459951 Ki = 0.18 nM T47768 CE2VA0 71459952 Ki = 0.39 nM T47768 CBHT09 71459962 EC50 = 0.6 nM T47768 C6NOP7 71459993 IC50 = 1670 nM T47768 CO2P3B 71460726 Ki = 3700 nM T47768 C12KHQ 71460850 Ki = 2.07 nM T47768 CJ65RV 71460942 Ki = 0.66 nM T47768 CC25XY 71460943 Ki = 4.69 nM T47768 CT52OM 71460944 Ki = 0.54 nM T47768 C6NLR9 71460945 Ki = 1.43 nM T47768 CBEV63 71461579 Ki = 118 nM T47768 CV60JN 71461663 Ki = 11.8 nM T47768 CFHE81 71461664 Ki = 0.87 nM T47768 CXT37B 71461665 Ki = 0.25 nM T47768 CY28RA 71461666 Ki = 0.25 nM T47768 C3O5EC 71461667 EC50 > 1000 nM T47768 C9Q6GY 71461668 Ki = 4.91 nM T47768 CD4Q0A 71461673 EC50 = 4.85 nM T47768 C75JTH 71462114 Ki = 132 nM T47768 C6H5QB 71462451 Ki = 760 nM T47768 C6N1FP 71462554 Ki = 0.6 nM T47768 C4ZD8G 71462655 Ki = 8.42 nM T47768 CB3L8W 71462656 Ki = 192 nM T47768 C1Y9IC 71463063 Ki = 2137 nM T47768 C2I5MZ 71463280 Ki = 0.12 nM T47768 CW8ZV5 71509717 EC50 = 5.9 nM T47768 CI21UZ 71605072 IC50 = 0.7079 nM T47768 C8D1CB 71605418 EC50 = 0.0397 nM T47768 CJ8GA4 71605419 EC50 = 0.00853 nM T47768 CT3YS1 71605420 EC50 = 0.057 nM T47768 C4UG0T 71605421 EC50 = 0.0933 nM T47768 C9Z7AT 71605588 EC50 = 0.0000912 nM T47768 CG8ZD6 71605589 EC50 = 0.000042 nM T47768 CU53FL 71605755 EC50 = 0.000107 nM T47768 CMZ8F3 71605756 EC50 = 0.000109 nM T47768 CIW95L 71613507 Ki > 10000 nM T47768 C26ORE 71613508 Ki > 10000 nM T47768 CHI7D3 71613509 Ki > 10000 nM T47768 CEO5Z2 71613709 Ki > 10000 nM T47768 C8X6TP 71613710 Ki > 10000 nM T47768 C82MIG 71613711 Ki = 5012 nM T47768 C0MC1V 71613712 Ki > 10000 nM T47768 CVC5H1 71613903 Ki = 4570 nM T47768 CX9PM4 71613904 Ki > 10000 nM T47768 C2BOG7 71613905 Ki = 711 nM T47768 CAJ61F 71613906 Ki = 724 nM T47768 CS3CN1 71613907 Ki > 10000 nM T47768 C0B7LC 71624265 Ki = 5.39 nM T47768 C7Q9VU 71624266 Ki = 16.13 nM T47768 CD9IO8 71624267 Ki = 533 nM T47768 CXZ6E1 71624268 Ki = 3.44 nM T47768 C0O6IR 71624269 Ki = 2.34 nM T47768 CW2G0T 71624270 Ki = 3.62 nM T47768 CBM1C8 71624387 Ki = 10.49 nM T47768 CML7K2 71624388 Ki = 16.26 nM T47768 C1B9VM 71624389 Ki = 23.27 nM T47768 C1A9BS 71660039 Ki = 60 nM T47768 CE0AX8 71660040 Ki = 165 nM T47768 CE5J8U 71660041 Ki = 45 nM T47768 CF4NS6 71660042 Ki = 28 nM T47768 CWBH85 71660081 Ki = 425 nM T47768 CWKO96 71660082 Ki = 84 nM T47768 CXZ1D7 71660083 Ki = 97 nM T47768 CJK9R5 71660084 Ki = 91 nM T47768 C7R1TA 71660085 Ki = 166 nM T47768 C4U5ZF 71660086 Ki = 96 nM T47768 C64TPF 71660087 Ki = 9 nM T47768 CM6I2K 71660088 Ki = 49 nM T47768 CD9CN8 71660125 Ki = 22 nM T47768 CDS7T3 71660126 Ki = 7 nM T47768 C1AIY3 71660127 Ki = 8 nM T47768 CJ43VK 71660128 Ki = 5 nM T47768 CF57LR 71660129 Ki = 23 nM T47768 C58SAC 71660130 Ki = 174 nM T47768 CG7UJ9 71660163 Ki = 16 nM T47768 CI0GU8 71660496 IC50 > 48500 nM T47768 C5XM1H 71680922 Ki = 1.51 nM T47768 CUW3Z8 71680923 Ki = 0.75 nM T47768 CWSC46 71680924 Ki = 0.82 nM T47768 CP5FK9 71681076 Ki = 3.5 nM T47768 C4LV9A 71681077 Ki = 9.09 nM T47768 CE0YC8 71681078 Ki = 1.13 nM T47768 CU57ZQ 71681079 Ki = 6.22 nM T47768 CW0MV2 71716116 Ki = 540 nM T47768 CVM39A 71716193 IC50 > 30000 nM T47768 CT82XD 71717930 Ki = 3 nM T47768 C8QO1W 71719108 Ki = 323 nM T47768 CZ8CL2 71719454 EC50 = 0.000516 nM T47768 C3LUG2 71720208 Ki = 39.2 nM T47768 CY89EO 71720682 EC50 = 0.00013 nM T47768 CCB3X2 71726555 Ki = 6.6 nM T47768 C4G5IU 71726685 Ki = 13 nM T47768 CLBE62 71726686 Ki = 9.3 nM T47768 CU47GC 71751564 Ki = 0.2 nM T47768 C0L7TE 71769137 Ki = 2300 nM T47768 CTX84S 71769138 Ki = 4200 nM T47768 C3YAR9 71769139 Ki > 10000 nM T47768 CWK9E7 71769267 Ki = 1600 nM T47768 C7G3EX 71769268 Ki > 10000 nM T47768 CEZW27 71769269 Ki = 3100 nM T47768 CW95UP 71819400 EC50 = 2000 nM T47768 C0EBP2 71819401 EC50 = 20 nM T47768 C7SQL1 71819402 EC50 = 16000 nM T47768 C8HK9Y 71819403 EC50 = 16000 nM T47768 C2MD4G 71819404 EC50 = 40000 nM T47768 CW0YD6 71819525 EC50 = 3200 nM T47768 CI4CE3 71819526 EC50 = 5000 nM T47768 CRF37P 71887675 Ki = 42 nM T47768 C0XHE7 72151344 Ki = 3040 nM T47768 C2QS5M 72153748 Ki > 100000 nM T47768 C7W2PU 72163557 Ki = 21 nM T47768 CMZ9E5 72163689 Ki = 14 nM T47768 CVJC81 72163691 Ki = 5.5 nM T47768 C4MA6E 72163693 Ki = 3.3 nM T47768 CZM45H 72163695 Ki = 20 nM T47768 C05KYU 72163804 Ki = 19 nM T47768 CS4RF2 72163806 Ki = 101 nM T47768 C2R0DE 72164175 IC50 = 23.7 nM T47768 CQHB67 72202465 Ki = 66 nM T47768 CZQ86Y 72374835 Ki = 22 nM T47768 CAK42B 72374836 Ki = 10.4 nM T47768 CWH6T3 72548703 IC50 = 1.1 nM T47768 C7NB1W 72711408 Ki = 0.085 nM T47768 C89COK 72711409 Ki = 6.6 nM T47768 C7FI6P 72711410 Ki = 9.6 nM T47768 CGZH63 72711945 EC50 = 10000 nM T47768 CE10DS 72711948 EC50 = 251.19 nM T47768 CY6GU0 72711950 EC50 = 79.43 nM T47768 CK7GI4 72711952 EC50 = 398.11 nM T47768 C3HFI1 72711954 EC50 = 1000 nM T47768 CLS1E3 72712149 EC50 = 501.19 nM T47768 CZ04MG 72712151 EC50 = 3162.28 nM T47768 C4M5SD 72712153 EC50 = 50.12 nM T47768 C3EIH2 72712155 EC50 = 10 nM T47768 CF5EX2 72712157 EC50 = 2.512 nM T47768 CO8PK5 72712368 EC50 = 794.33 nM T47768 C29YGC 72712370 EC50 = 15.85 nM T47768 C0ILU3 72712589 EC50 = 12.59 nM T47768 CRC5V0 72712592 EC50 = 31.62 nM T47768 C9O4MK 72712594 EC50 = 6.31 nM T47768 C19NWJ 72712596 EC50 = 5.012 nM T47768 C0EI8T 72712793 EC50 = 15.85 nM T47768 CUZE98 72712795 EC50 = 50.12 nM T47768 COYH24 72712797 EC50 = 25.12 nM T47768 C3C1GQ 72712799 EC50 = 5.012 nM T47768 CE4NJ7 72712801 EC50 = 31.62 nM T47768 CYEJ30 72713098 Ki = 0.371 nM T47768 CJT7L9 72713099 Ki = 3.35 nM T47768 C4MWE1 72713100 Ki = 1.66 nM T47768 CPY8F1 72713101 Ki = 7.55 nM T47768 CBVG86 72713102 Ki = 0.28 nM T47768 C6WO0U 72713103 EC50 = 60 nM T47768 CLRX12 72713104 Ki = 0.43 nM T47768 CF1U5Z 72713191 EC50 = 12.59 nM T47768 C67REA 72713193 EC50 = 630.96 nM T47768 CC6Q5R 72771081 Ki < 100 nM T47768 CRK2J6 73212901 EC50 >= 10000 nM T47768 CC65OA 73213195 Ki > 10000 nM T47768 CW83DK 73213196 Ki > 10000 nM T47768 COL97Y 73295685 IC50 = 343 nM T47768 CNA8O3 73345364 Ki = 2340 nM T47768 CMU18J 73345366 Ki = 6200 nM T47768 C7ZN1K 73345634 Ki = 354.81 nM T47768 C4NHU9 73346590 EC50 = 39.81 nM T47768 CY03SQ 73346599 Ki = 54.8 nM T47768 CU7C6J 73346891 Ki = 2750 nM T47768 CS5F3B 73347271 Ki = 0.5 nM T47768 CQJ36Z 73347341 Ki > 10000 nM T47768 CH2T1I 73347643 Ki = 23 nM T47768 C5HXL6 73347644 Ki = 52 nM T47768 C46QVZ 73348688 Ki = 5880 nM T47768 CM70YA 73349151 Ki = 4.92 nM T47768 C9Z3KC 73349647 Ki = 24.8 nM T47768 C80THJ 73350137 Ki > 4500 nM T47768 CN5S4A 73350483 Ki = 79.9 nM T47768 C5GAW0 73351393 EC50 = 15 nM T47768 CWA73N 73352217 Ki = 2.23 nM T47768 CL2W3H 73352233 Ki = 7.2 nM T47768 CSY9E4 73352234 EC50 = 3200 nM T47768 C7D1LF 73352661 Ki = 33.2 nM T47768 CKFA02 73353693 Ki = 1.49 nM T47768 C2VQJ1 73354161 EC50 = 501.19 nM T47768 CO3ZS7 73354458 Ki = 1660 nM T47768 C0SBM2 73354619 Ki > 4500 nM T47768 COS31U 73354624 Ki = 368 nM T47768 C2HJ6O 73355223 Ki = 0.9 nM T47768 C3Z5LT 73355419 Ki = 2125 nM T47768 C3Q9FB 73356023 Ki = 15100 nM T47768 C83ZPI 73356767 Ki = 4 nM T47768 CJT8Y2 73356768 Ki = 40 nM T47768 C2E7QW 75201901 Ki = 8200 nM T47768 CJQ25A 76309739 Ki = 52 nM T47768 CC01JG 76309740 Ki = 71 nM T47768 C2LZD4 76309826 Ki = 0.3 nM T47768 CB78KL 76309827 Ki = 0.14 nM T47768 C68BLJ 76309828 Ki = 1.59 nM T47768 C69JCU 76313421 Ki = 205 nM T47768 CJR57Q 76313422 Ki = 1315 nM T47768 CP3HV7 76313424 Ki = 601 nM T47768 CU56FN 76313425 Ki = 284 nM T47768 CPJ4N3 76313426 Ki = 447 nM T47768 C7LV2A 76313427 Ki = 46 nM T47768 C35USC 76313542 Ki = 0.75 nM T47768 C6J2WF 76313543 Ki = 0.82 nM T47768 CZSU65 76313544 Ki = 9.09 nM T47768 CTN6G1 76316935 Ki = 143 nM T47768 C1AW8J 76316936 Ki = 133 nM T47768 C1GU9H 76317053 Ki = 2.69 nM T47768 CM9RC0 76317054 Ki = 4.34 nM T47768 CSYN97 76317055 Ki = 1.13 nM T47768 C0SWX7 76317056 Ki = 0.32 nM T47768 CP95SN 76317057 Ki = 1.44 nM T47768 CF83DA 76320665 Ki = 312 nM T47768 C5W1XJ 76320666 Ki = 190 nM T47768 CPKY85 76320762 Ki = 5.58 nM T47768 C0MI1G 76324308 Ki = 85 nM T47768 CI2A6W 76324309 Ki = 153 nM T47768 CT9XB8 76324310 Ki = 26 nM T47768 C4QM6R 76324311 Ki = 265 nM T47768 CG9MB3 76324401 Ki = 0.14 nM T47768 CU12ZJ 76324412 Ki = 1.61 nM T47768 C6AY5S 76327872 Ki = 468 nM T47768 CL58DY 76327874 Ki = 74 nM T47768 CBVL29 76327875 Ki = 367 nM T47768 C64JDN 76327876 Ki = 209 nM T47768 C3G1LA 76327877 Ki = 840 nM T47768 CIX43W 76327982 Ki = 123.2 nM T47768 CCN1M9 76331524 Ki = 481 nM T47768 CQ35XY 76331525 EC50 = 1563 nM T47768 CLU90M 76331610 IC50 = 1.8 nM T47768 CB4JI7 76331634 Ki = 225.3 nM T47768 CCW07O 76331635 Ki = 1.51 nM T47768 CRA1Y0 76331636 Ki = 6.22 nM T47768 CKZ7T2 76335142 Ki = 348 nM T47768 CQKT47 76335143 Ki = 343 nM T47768 C6K5RY 76335144 Ki = 741 nM T47768 CECO35 76335145 Ki = 961 nM T47768 C6F1BS 76335253 Ki = 3.5 nM T47768 COK40D 76335254 Ki = 0.29 nM T47768 CZP08R 76335255 Ki = 68.4 nM T47768 CM27VY 78210001 Ki = 3.2 nM T47768 CTI5S8 81689720 Ki = 112 nM T47768 C3WU0Y 85937411 EC50 > 100000 nM T47768 CGH7J9 86279209 Ki = 8.19 nM T47768 C5C9KE 86648372 Ki = 1775 nM T47768 CG1UD2 89001045 Ki = 56.45 nM T47768 C97GYK 89435126 Ki = 0.726 nM T47768 CL5R0T 89435196 Ki = 0.813 nM T47768 C7X1VI 89435275 Ki = 0.953 nM T47768 C08YSC 89435280 Ki = 0.826 nM T47768 CI67KS 89702731 IC50 = 40 nM T47768 CZSC16 90306849 Ki = 0.82 nM T47768 C03HOW 90392373 Ki = 0.627 nM T47768 C0OAE4 90392376 Ki = 3.44 nM T47768 C47BLH 90397724 Ki = 0.578 nM T47768 C54EUB 90644257 Ki = 415 nM T47768 CZ10JE 90644258 Ki = 76.3 nM T47768 CV7U4P 90644259 Ki = 3.06 nM T47768 CGN7C6 90644461 IC50 = 21900 nM T47768 CI2TV6 90644873 Ki = 0.24 nM T47768 C3WD0A 90644874 Ki = 0.24 nM T47768 CGBL95 90644875 Ki = 0.1 nM T47768 C9B0JT 90645382 IC50 > 1000 nM T47768 C3VIY8 90645383 IC50 > 1000 nM T47768 C6YPT9 90645384 IC50 > 1000 nM T47768 CPB25R 90645385 IC50 > 1000 nM T47768 C18HBT 90645386 IC50 > 1000 nM T47768 C1DOG7 90654745 Ki > 375 nM T47768 CX3WT1 90654746 Ki > 375 nM T47768 CC70MH 90654747 Ki > 375 nM T47768 C4ZQD5 90654748 Ki > 375 nM T47768 CBV23K 90654749 Ki > 375 nM T47768 C87NYV 90654750 Ki > 375 nM T47768 C20FOK 90654751 Ki > 375 nM T47768 CT91LC 90654752 Ki > 375 nM T47768 C1Y6QN 90655511 EC50 = 6.3 nM T47768 CCM78A 90655513 EC50 = 18.6 nM T47768 CIQV28 90655825 EC50 = 223 nM T47768 C6V1PS 90655826 EC50 = 2.7 nM T47768 CNPC03 90655827 EC50 = 2.3 nM T47768 CFAZ39 90655828 EC50 = 1.2 nM T47768 C63YPH 90655829 EC50 = 2.1 nM T47768 C7C5BM 90655970 Ki = 167.8 nM T47768 CTV50C 90655971 Ki = 41.5 nM T47768 C1S5UB 90655972 Ki = 30.3 nM T47768 CV6A5T 90655973 Ki = 1.46 nM T47768 CL0D4Y 90655974 Ki = 1.05 nM T47768 C51CQN 90655975 Ki = 10.6 nM T47768 C2USA9 90655976 Ki = 1.97 nM T47768 CLKW80 90655977 Ki = 100 nM T47768 C96DUE 90655978 Ki = 10.2 nM T47768 C1N5QA 90655979 Ki = 33.4 nM T47768 C6FN2S 90656087 Ki = 186 nM T47768 C2QY3H 90656088 Ki = 6.55 nM T47768 CW2P5Q 90656089 Ki = 26.5 nM T47768 C8TV7C 90656090 EC50 = 130000 nM T47768 CWE5X6 90656115 IC50 = 8200 nM T47768 CK9FP8 90656664 Ki = 3.2 nM T47768 CC6LY3 90656665 EC50 = 2.75 nM T47768 COGW86 90656666 Ki = 4 nM T47768 C9YKV8 90656667 Ki = 4.2 nM T47768 C3WLH8 90656668 Ki = 1 nM T47768 CP1ZW6 90663949 Ki > 5000 nM T47768 CZ9GL5 90663950 Ki = 85 nM T47768 CFK27M 90663951 Ki = 833 nM T47768 CBT6F1 90663952 Ki > 5000 nM T47768 C1QAB3 90663953 Ki = 53 nM T47768 CPNS27 90664349 Ki = 0.43 nM T47768 C0I6XM 90664791 Ki = 310 nM T47768 C3QA8Z 90664881 EC50 = 19.5 nM T47768 C4US3O 90664914 Ki = 330 nM T47768 C9Z0DQ 90665047 Ki = 270 nM T47768 C5VZC6 90666479 Ki = 0.16 nM T47768 CV1XD0 90666576 Ki = 9.2 nM T47768 C2NG3A 90666726 Ki > 10000 nM T47768 C5DG9V 90666727 Ki > 10000 nM T47768 C26HUP 90666728 Ki > 10000 nM T47768 CK0W6U 90666729 Ki > 10000 nM T47768 CM75TG 90666730 Ki = 777 nM T47768 C4D6WT 90666731 Ki > 5800 nM T47768 C0GWK7 90666732 Ki > 3000 nM T47768 CT70RV 90666733 Ki = 3523 nM T47768 CT0O1B 90666734 Ki > 10000 nM T47768 CCUK67 90666735 Ki = 1540 nM T47768 CWI2S7 90666736 Ki > 3000 nM T47768 C0BNE6 90667279 Ki = 830 nM T47768 CWOB91 90667280 Ki > 890 nM T47768 CU2XP8 91801212 EC50 = 57.6 nM T47768 CR93LZ 91928491 Ki = 38 nM T47768 C2UZ4P 91928492 Ki = 63 nM T47768 CK4U6G 93967682 Ki = 478 nM T47768 COM0Q7 94156776 Ki = 2430 nM T47768 C7GBD9 94438674 EC50 = 4.6 nM T47768 CMI13V 95177310 Ki = 45700 nM T47768 CA2LJ1 95241239 Ki = 2.5 nM T47768 CSPX47 95261164 Ki = 6920 nM T47768 C98WTN 95265878 Ki = 2470 nM T47768 C0KVB7 99941396 EC50 = 10000 nM T47768 CCY0O2 100951644 IC50 = 60000 nM T47768 C07VRA 101341769 Ki = 3150 nM T47768 CW3LH2 101882818 Ki = 3.39 nM T47768 CW5H9D 101882819 Ki = 201 nM T47768 CGQV37 101882820 Ki > 5000 nM T47768 CNHS29 101898709 EC50 = 41 nM T47768 CJX06V 101910788 EC50 >= 10000 nM T47768 CB5DK1 102004349 Ki = 7 nM T47768 CPT9B3 102269996 Ki = 0.42 nM T47768 C9T1NI 102269998 Ki = 0.56 nM T47768 COFT20 102270003 Ki = 0.29 nM T47768 CR4KN5 102270004 Ki = 3 nM T47768 CP5F4Q 102270005 Ki = 12.8 nM T47768 C3FX4P 102270006 Ki = 2.03 nM T47768 CFA7K6 102270007 Ki = 2.37 nM T47768 CD19TA 102270008 Ki = 1.23 nM T47768 CS7V1U 114284704 EC50 = 6800 nM T47768 C0BCI6 117705988 EC50 = 5.3 nM T47768 CEP48V 117706009 Ki = 0.308 nM T47768 CMO27R 117706010 Ki = 1.56 nM T47768 C67SPE 117706054 Ki = 0.545 nM T47768 C12FIV 117706085 Ki = 2.5 nM T47768 CWU50D 117738965 IC50 = 2728 nM T47768 CSJ3H4 117860306 EC50 = 22 nM T47768 C3A7QZ 118200491 Ki = 30.3 nM T47768 CR52EZ 118200640 Ki = 49.3 nM T47768 CUCJ65 118263805 IC50 = 79 nM T47768 C9JV1T 118263857 IC50 = 183 nM T47768 CRY49P 118263892 IC50 = 176 nM T47768 C9YVS2 118263923 IC50 = 4390 nM T47768 C5HCS3 118264001 IC50 = 829 nM T47768 C38LHY 118264112 IC50 = 31.1 nM T47768 C5CDE0 118562359 Ki = 49 nM T47768 CS63OE 118562362 Ki = 46 nM T47768 CWH9B5 118562372 Ki = 117 nM T47768 C60BSA 118562375 EC50 = 0.2 nM T47768 CE3D0A 118562384 EC50 = 4 nM T47768 C7IVW9 118562402 Ki = 262 nM T47768 C63EGC 118562428 EC50 > 1000 nM T47768 CE53DJ 118562440 Ki = 10 nM T47768 CW26NV 118562451 Ki = 69 nM T47768 C7G5HO 118562469 Ki = 92 nM T47768 C3BIL8 118562502 Ki = 304 nM T47768 C5JKQ9 118562510 EC50 = 1 nM T47768 C12CKV 118562522 EC50 > 1000 nM T47768 CF6LK7 118562538 EC50 = 11 nM T47768 C6FOS9 118562556 Ki = 126 nM T47768 C25MXS 118562567 Ki = 19 nM T47768 C3TQE7 118562573 EC50 > 1000 nM T47768 CJF1E6 118562576 Ki = 40 nM T47768 C5QB2S 118562584 Ki = 8 nM T47768 C6TC3D 118562598 Ki = 90 nM T47768 CWA4B2 118562606 Ki = 3 nM T47768 C0XIN5 118567313 Ki = 13 nM T47768 C6PA1C 118567531 Ki = 34 nM T47768 CD4XK8 118567534 Ki = 261 nM T47768 CLVO18 118567538 EC50 = 25 nM T47768 C1CP6Z 118567543 Ki = 175 nM T47768 C32PGF 118567545 Ki = 123 nM T47768 C7G8IT 118567547 Ki = 204 nM T47768 CN1DU3 118567549 Ki = 636 nM T47768 CKQ15C 118567550 Ki = 606 nM T47768 CJ43GO 118567552 Ki = 727 nM T47768 CV7U9Y 118567593 EC50 > 1000 nM T47768 CXW0K9 118567604 EC50 = 4 nM T47768 C4ULH8 118567605 Ki = 304 nM T47768 C7DO6S 118567606 Ki = 930 nM T47768 C8TP7C 118567608 EC50 = 1 nM T47768 C70RDE 118567618 Ki = 535 nM T47768 CGN3Z4 118567654 Ki = 534 nM T47768 CJOK48 118567670 Ki = 437 nM T47768 C4GDV1 118567672 Ki = 516 nM T47768 CK5T2Z 118567678 EC50 > 1000 nM T47768 CCY60Z 118567689 Ki = 127 nM T47768 C59GUQ 118567742 EC50 > 1000 nM T47768 C36JSR 118567743 Ki = 90 nM T47768 C5NI2E 118567744 Ki = 57 nM T47768 CI0JY2 118567747 Ki = 93 nM T47768 CBM3Q5 118662014 Ki = 26 nM T47768 CK8Y3E 118662042 Ki = 4.5 nM T47768 CS81PR 118662074 Ki = 1.14 nM T47768 C8AF6I 118662117 Ki = 4 nM T47768 CBJ16O 118662129 Ki = 230 nM T47768 C4ZP0L 118662159 Ki = 1.2 nM T47768 CR6IU7 118662169 Ki = 1590 nM T47768 C7VE1O 118662183 Ki = 170 nM T47768 C1VR3B 118662189 Ki = 1 nM T47768 CG0R6H 118662291 Ki = 2.8 nM T47768 CI17PS 118662309 Ki = 30.5 nM T47768 CCIP14 118662342 Ki = 0.4 nM T47768 CB79UC 118662456 Ki = 3.5 nM T47768 C5LZ8I 118662460 Ki = 0.6 nM T47768 CM8TB4 118705898 Ki = 0.18 nM T47768 C6RW0E 118705901 Ki = 0.11 nM T47768 C8ZM3D 118709349 Ki = 314 nM T47768 C58BHC 118709350 Ki = 426 nM T47768 CBU7N4 118709351 Ki > 100000 nM T47768 CE7X1W 118709352 Ki > 100000 nM T47768 C9FAV4 118709353 Ki = 5.7 nM T47768 CSY8D4 118709354 Ki = 20.8 nM T47768 CSBQ79 118709355 Ki > 100000 nM T47768 C01ZSF 118709356 Ki = 114 nM T47768 CK3S0G 118709357 Ki = 190 nM T47768 CIJX58 118709358 Ki = 51.9 nM T47768 CT0F3M 118709359 Ki > 100000 nM T47768 CN3UC7 118709360 Ki = 4.03 nM T47768 CW32LQ 118710801 Ki = 4300 nM T47768 CQ6O7Y 118710802 Ki = 6000 nM T47768 CP3WR9 118710803 Ki = 4400 nM T47768 C27YCZ 118710804 Ki = 3620 nM T47768 CS9X1P 118710805 Ki = 4450 nM T47768 C0O5KT 118710807 Ki = 6000 nM T47768 CHU9L5 118711127 EC50 = 19000 nM T47768 CHC14P 118711128 EC50 = 30200 nM T47768 CBR9W6 118711129 EC50 = 370 nM T47768 CO31BE 118711130 EC50 = 8900 nM T47768 CR38FY 118711131 EC50 = 10000 nM T47768 CQX8H5 118711132 EC50 = 370 nM T47768 CAXH38 118711133 EC50 = 10300 nM T47768 CI1QT3 118711134 EC50 = 41 nM T47768 C4MRB0 118711135 EC50 = 41 nM T47768 CGMW34 118711136 EC50 = 13600 nM T47768 C6HCN7 118711137 EC50 = 1540 nM T47768 C3DVF8 118711138 EC50 = 370 nM T47768 CP6WQ1 118711209 EC50 = 100 nM T47768 CV85YO 118711243 Ki = 2.1 nM T47768 CKUT03 118711485 Ki = 0.3 nM T47768 CMY0F1 118711490 Ki = 0.24 nM T47768 CMRV59 118711491 Ki = 0.36 nM T47768 CL9F4B 118711887 Ki = 7.7 nM T47768 CBK60I 118713122 Ki = 979 nM T47768 C5J0UN 118713123 Ki = 284 nM T47768 CJ38GQ 118713124 Ki = 362 nM T47768 CCIS67 118713125 Ki = 540 nM T47768 CDU9H7 118713126 Ki = 1441 nM T47768 C8TPM0 118713127 Ki > 10000 nM T47768 C9E8OS 118713128 Ki = 439 nM T47768 CRVW31 118713129 Ki = 52 nM T47768 CO8UJ6 118713130 Ki > 10000 nM T47768 CL25HD 118713131 Ki > 10000 nM T47768 CI52KQ 118713132 Ki > 10000 nM T47768 C5MJX6 118713133 Ki > 10000 nM T47768 C4MHO8 118713134 Ki > 10000 nM T47768 CT7EU4 118713135 Ki = 2820 nM T47768 CZFQ32 118713136 Ki > 10000 nM T47768 C0P3QL 118713137 Ki > 10000 nM T47768 CE4Z7B 118713138 Ki > 10000 nM T47768 C14HFW 118713139 Ki > 10000 nM T47768 C7HO5D 118713140 Ki > 10000 nM T47768 C7NHP9 118713141 Ki = 334 nM T47768 CUY58S 118713142 Ki = 18 nM T47768 C78LKO 118716009 EC50 = 0.4 nM T47768 C5BJA6 118716010 EC50 = 1.09 nM T47768 C9BFP5 118718265 Ki = 374 nM T47768 CS14YZ 118718266 Ki = 785 nM T47768 CPC23W 118718272 Ki = 1284 nM T47768 C2Y4PK 118718273 Ki = 3976 nM T47768 C8FC1Q 118718274 Ki = 251 nM T47768 CJZ1F7 118718276 Ki = 1414 nM T47768 CCFR52 118718277 Ki = 782 nM T47768 CC0KE5 118718279 Ki = 617 nM T47768 CK1Q9B 118718280 Ki = 442 nM T47768 CDH69C 118718284 Ki = 758 nM T47768 CLRD02 118718285 Ki = 3447 nM T47768 CYI4T2 118718286 Ki = 752 nM T47768 CA9N0S 118718288 Ki = 123 nM T47768 CVT94Z 118718289 Ki = 674 nM T47768 C1RAX5 118718290 Ki = 566 nM T47768 CKNL94 118718291 Ki = 1486 nM T47768 CKN54J 118718292 Ki = 905 nM T47768 CC6U5D 118718293 Ki = 2620 nM T47768 C64JUV 118718294 Ki = 4169 nM T47768 CZMR06 118718296 Ki = 2106 nM T47768 C92CER 118718297 Ki = 2407 nM T47768 CP23YE 118718298 Ki = 1204 nM T47768 COA69M 118718299 Ki = 1706 nM T47768 CSW82H 118718300 Ki = 998 nM T47768 C2EGJ8 118718301 Ki = 1336 nM T47768 CO5BV4 118718302 Ki = 458 nM T47768 C29GAH 118719100 Ki > 4500 nM T47768 CU10SI 118722557 Ki = 13.2 nM T47768 CTF9L6 118722880 Ki = 11 nM T47768 CDI8J1 118722882 Ki = 22 nM T47768 CA51CQ 118724536 Ki > 5000 nM T47768 CH4LB0 118724977 Ki > 5000 nM T47768 C9SN0M 118724979 Ki = 2022 nM T47768 CH9GT5 118724980 Ki = 688 nM T47768 CG7SQ8 118724984 Ki > 5000 nM T47768 C29CVM 118725741 EC50 = 2400 nM T47768 C0HM6Y 118725745 EC50 = 7800 nM T47768 CXL16I 118725841 EC50 = 1800 nM T47768 C49YCX 118725843 EC50 = 100000 nM T47768 CCQ85P 118725848 EC50 = 3300 nM T47768 C1Q5IB 118725849 EC50 = 100000 nM T47768 CE86DJ 118725850 EC50 = 6800 nM T47768 CBDA90 118725853 EC50 = 255 nM T47768 CET5Y3 118725854 EC50 = 3800 nM T47768 C2LA6F 118725855 EC50 = 150 nM T47768 CO8B9L 118725856 EC50 = 1750 nM T47768 CMO86W 118725857 EC50 = 52500 nM T47768 C61VHK 118725858 EC50 = 34500 nM T47768 C3T8YZ 118726261 IC50 = 29 nM T47768 C6I5HS 118726262 IC50 = 110 nM T47768 C10BIV 118726263 IC50 = 36 nM T47768 CA43CF 118726264 IC50 = 47 nM T47768 CLSG96 118726265 IC50 = 29 nM T47768 CYL40S 118726266 IC50 = 80 nM T47768 CPR0K2 118726267 IC50 = 69 nM T47768 CH9A3M 118726268 IC50 = 103 nM T47768 CEH89Y 118726269 IC50 = 79 nM T47768 CT7H2M 118726270 IC50 = 57 nM T47768 C1UD6R 118726271 IC50 = 990 nM T47768 CRK62Y 118726272 IC50 = 540 nM T47768 CF25IA 118726273 IC50 = 820 nM T47768 CFNX71 118726846 Ki = 13.23 nM T47768 C5LUM4 118726847 Ki = 19.61 nM T47768 C5MSK4 118726848 Ki = 63.08 nM T47768 CT0O1J 118726849 Ki = 57.52 nM T47768 CQH1G3 118731120 EC50 = 0.1 nM T47768 CDN86Z 118731405 Ki = 14 nM T47768 CK5W7M 118731406 Ki = 47 nM T47768 C29ESD 118731407 Ki = 17 nM T47768 CAP48T 118731408 Ki = 73 nM T47768 C12NJU 118731409 Ki = 27 nM T47768 CM06BI 118731410 Ki = 53 nM T47768 CP84KM 118731411 Ki = 13 nM T47768 C5MK1D 118731412 Ki = 351 nM T47768 CPD5R9 118731413 Ki = 93 nM T47768 CY9NH0 118731414 Ki = 7.7 nM T47768 CR6K5D 118731415 Ki = 12 nM T47768 CMR93J 118731416 Ki = 10.1 nM T47768 CQ39OA 118731417 Ki = 80 nM T47768 CK76UL 118731418 Ki = 3.8 nM T47768 CRXY76 118731419 Ki = 14 nM T47768 C9A4RX 118731420 Ki = 294 nM T47768 C3N0VC 118731422 Ki = 38 nM T47768 C4FT8K 118731423 Ki = 5.6 nM T47768 C1L4QH 118731424 Ki = 4.2 nM T47768 CB0R9K 118731425 Ki = 5.8 nM T47768 CW35DR 118731426 Ki = 3.1 nM T47768 CP61XB 118731427 Ki = 3.9 nM T47768 CD51ZQ 118731428 Ki = 159 nM T47768 CNT5W9 118737392 EC50 = 7000 nM T47768 CUT4V5 118737393 EC50 > 10000 nM T47768 CT24GR 118737394 EC50 > 10000 nM T47768 C19VKC 118737395 EC50 = 3000 nM T47768 CSL4C7 118737396 EC50 = 2000 nM T47768 C59YKQ 118737397 EC50 = 5000 nM T47768 C5SAR8 118737398 EC50 = 10000 nM T47768 CR1L6M 118737399 EC50 > 10000 nM T47768 CWO42N 121365644 Ki > 10000 nM T47768 CG52CR 121365655 Ki = 8170 nM T47768 C9ND2K 121373679 Ki = 1749 nM T47768 C0J9GQ 121432154 Ki = 0.2512 nM T47768 C1LIT9 121596705 Ki = 1.1 nM T47768 CO9A8T 121614380 EC50 = 860 nM T47768 C85NKZ 121614424 EC50 = 660 nM T47768 CP1D8B 121614426 EC50 = 370 nM T47768 CSRW32 121614490 Ki = 36.4 nM T47768 C6KIU4 121614638 EC50 = 370 nM T47768 CC3E1H 121614661 EC50 = 370 nM T47768 CRUE82 121614715 Ki = 6.47 nM T47768 CRN4D5 121614717 EC50 = 8910 nM T47768 C9R6HA 121614780 EC50 = 3310 nM T47768 CQ3LD2 121614853 Ki = 4.65 nM T47768 CLC5E9 121661888 EC50 = 4020 nM T47768 CYI9H2 121661890 EC50 = 8080 nM T47768 CRY9A8 121684957 EC50 = 1120 nM T47768 CWP9E2 122178420 EC50 = 6.31 nM T47768 CQ7YP3 122178421 EC50 = 5.248 nM T47768 C5QZT2 122178422 EC50 = 2.512 nM T47768 C74MRY 122178423 EC50 = 5.129 nM T47768 C5JCY2 122178425 EC50 = 2.754 nM T47768 C1A2JB 122178426 EC50 = 1.66 nM T47768 CMH98S 122178427 EC50 = 6.761 nM T47768 CRKB15 122179557 EC50 = 2.57 nM T47768 C8OF5S 122179558 EC50 = 4.074 nM T47768 C93YZC 122179560 EC50 = 3.236 nM T47768 C3UV6A 122182776 Ki = 788 nM T47768 CVMP98 122182777 Ki = 133 nM T47768 C20HCF 122182778 Ki = 675 nM T47768 C3S5RY 122182780 Ki > 1000 nM T47768 C18PTI 122182782 Ki > 1000 nM T47768 C6R8UI 122182784 Ki = 670 nM T47768 CG7N6Q 122182786 Ki = 123 nM T47768 CYJ34R 122182788 Ki = 422 nM T47768 CDJ0N9 122182790 Ki > 1000 nM T47768 CWYQ85 122182792 Ki > 1000 nM T47768 C80PUY 122183206 Ki = 4.8 nM T47768 C61ZWM 122183207 Ki = 8.8 nM T47768 CP7G1A 122183208 Ki = 3.2 nM T47768 C6GLF5 122183209 Ki = 5.6 nM T47768 CIP5Y3 122183210 Ki = 15 nM T47768 C9YU5A 122183211 Ki = 2.8 nM T47768 CIL5O7 122183212 Ki = 21 nM T47768 CMR9Q4 122183213 Ki = 0.24 nM T47768 CKP97B 122183214 Ki = 120 nM T47768 CWH04D 122183215 Ki = 1200 nM T47768 CULZ39 122183217 Ki = 5.2 nM T47768 C0CPO2 122183218 Ki = 5 nM T47768 CDUW32 122183219 Ki = 2.6 nM T47768 CA7R3L 122183220 Ki = 26 nM T47768 C7EO2T 122183221 Ki = 39 nM T47768 C7QKU8 122183222 Ki = 27 nM T47768 CA0B9X 122183223 Ki = 3.8 nM T47768 CXE52Q 122183281 Ki = 6.6 nM T47768 CV0FU5 122183282 Ki = 4.3 nM T47768 CEP3K5 122183283 Ki = 13 nM T47768 CB9Z1T 122183284 Ki = 1.4 nM T47768 CJ6RO8 122193596 IC50 > 10000 nM T47768 CS64OW 122194218 EC50 = 0.0629 nM T47768 CS1IN2 122194219 EC50 = 0.0643 nM T47768 CNE13U 122194668 Ki = 17.2 nM T47768 C5K8XH 122197315 IC50 = 404 nM T47768 CFWE98 122197316 IC50 = 764 nM T47768 CZ03XS 122197485 IC50 = 130 nM T47768 C0WTE6 122197486 IC50 = 120 nM T47768 C1TP0H 122197487 IC50 = 220 nM T47768 CSN3V4 122197488 IC50 = 103 nM T47768 C6LC2J 122197489 IC50 > 10000 nM T47768 CPCF21 122197490 IC50 = 44 nM T47768 CF8X5R 122197491 IC50 = 200 nM T47768 CMA83V 122197492 IC50 = 6.4 nM T47768 CX4I7N 122197493 IC50 = 16 nM T47768 CWZA97 122197494 IC50 = 420 nM T47768 CTKY87 122197495 IC50 = 2050 nM T47768 CH9O2Q 122197496 IC50 = 360 nM T47768 C5I8CM 122197497 IC50 = 59 nM T47768 C7EF4P 122197498 IC50 = 690 nM T47768 C1BDZ4 122197499 IC50 = 7 nM T47768 C7F8CK 122197500 IC50 > 9500 nM T47768 CMH7K2 122197501 IC50 > 10000 nM T47768 CD3L6S 122197502 IC50 > 10000 nM T47768 C7O1EP 122197503 IC50 = 690 nM T47768 CYE18M 122197504 IC50 = 53 nM T47768 C9W2FQ 122197505 IC50 = 56 nM T47768 C45VUL 122197506 IC50 = 160 nM T47768 CEP3J0 122197507 IC50 = 500 nM T47768 C9B5DC 122197508 IC50 = 1080 nM T47768 CZTO90 122197509 IC50 = 2000 nM T47768 C7SJO2 122197510 IC50 = 230 nM T47768 CH93LB 122197511 IC50 = 1030 nM T47768 CL78AV 122197512 IC50 = 82 nM T47768 CAQ5B0 122409965 Ki = 321 nM T47768 C0K8BS 122589938 Ki = 1065 nM T47768 CBU38O 122589952 Ki = 731 nM T47768 CTNU73 123445395 Ki = 0.83 nM T47768 C51MTO 124565311 Ki = 35 nM T47768 CK78QD 126619369 EC50 = 14000 nM T47768 C09XWQ 126619371 EC50 > 30000 nM T47768 CZT1F5 126619377 EC50 = 13300 nM T47768 CL60JG 126619380 EC50 = 8600 nM T47768 C2S5RA 126619383 EC50 > 30000 nM T47768 C9M0RG 126619391 EC50 = 3300 nM T47768 CJFZ14 126619393 EC50 = 6100 nM T47768 C3DJ4Q 126619396 EC50 = 4900 nM T47768 C45OHN 126619399 EC50 = 3300 nM T47768 C03QWD 126619400 EC50 = 13800 nM T47768 CBD9T4 126619405 EC50 > 30000 nM T47768 CN2T4V 126619407 EC50 = 8800 nM T47768 CMZP03 126619413 EC50 > 30000 nM T47768 C0BCH9 126619418 EC50 = 4200 nM T47768 CSDH62 126619420 EC50 = 2800 nM T47768 CN7A2T 126619428 EC50 = 3900 nM T47768 CZJ43A 126619429 EC50 = 10100 nM T47768 CR7Q3S 126619433 EC50 > 30000 nM T47768 CONM37 126619448 EC50 > 30000 nM T47768 C09PAE 126744799 Ki = 46 nM T47768 COJ60B 126744800 Ki = 144 nM T47768 C2U4GO 126744949 Ki = 190 nM T47768 C0FKA4 126744972 Ki = 11 nM T47768 C8OXG3 127024961 Ki = 1050 nM T47768 CZ5NJ7 127025173 Ki = 14 nM T47768 C9FBD2 127025219 Ki = 0.47 nM T47768 CL3VG1 127025528 Ki = 0.38 nM T47768 C5D7WM 127025817 Ki = 1.5 nM T47768 CTBN56 127026052 Ki < 10000 nM T47768 CKP92G 127026454 EC50 = 19.95 nM T47768 CI3YF5 127026455 EC50 = 11.48 nM T47768 CRDW90 127026456 EC50 = 5.623 nM T47768 CO5S0Z 127026457 EC50 = 3.631 nM T47768 C6D7EV 127028324 Ki = 0.94 nM T47768 CW6RV7 127028653 Ki = 0.042 nM T47768 CO7H8W 127029282 Ki = 1.71 nM T47768 CIW9F7 127029283 Ki = 3.3 nM T47768 C8AO1V 127029284 Ki = 0.5 nM T47768 C1YEA7 127030671 Ki > 450 nM T47768 CSK04O 127032208 Ki = 5.75 nM T47768 CR3TB5 127032209 Ki = 7.2 nM T47768 C2SP1T 127032210 EC50 = 11.6 nM T47768 CXJY65 127032211 Ki = 22 nM T47768 CK29CG 127032212 Ki = 5.81 nM T47768 CQ25BG 127032213 Ki = 4.61 nM T47768 CY72AX 127033106 Ki = 3480 nM T47768 CN0BZ9 127033398 Ki = 0.692 nM T47768 CFR46S 127033399 Ki = 24.7 nM T47768 C1HO7F 127033703 Ki > 450 nM T47768 CB12AP 127033704 Ki = 231 nM T47768 CML91J 127033967 EC50 = 19.2 nM T47768 C4NIU0 127034022 Ki = 49.1 nM T47768 C7ORD8 127034023 Ki = 289 nM T47768 CLR2J7 127034153 IC50 = 12000 nM T47768 CEWM81 127034292 Ki = 342 nM T47768 CBOC84 127034554 Ki = 108 nM T47768 CZ61LK 127034966 EC50 > 5011.87 nM T47768 CA0SN5 127034967 EC50 > 5011.87 nM T47768 CQ0ZT9 127035062 Ki = 341 nM T47768 CU49VE 127036186 Ki < 10000 nM T47768 CG06BD 127036932 Ki = 2818.38 nM T47768 CVW71O 127036953 Ki = 1737.8 nM T47768 CBL83N 127040383 IC50 = 70.4 nM T47768 C87QAX 127040384 IC50 = 24 nM T47768 C52QVR 127040385 IC50 = 677.8 nM T47768 CP7FE3 127041366 EC50 = 20.42 nM T47768 C9J2GY 127041367 EC50 = 398.11 nM T47768 CYN01M 127041368 EC50 = 4.677 nM T47768 C6E2AQ 127041630 IC50 = 2.3 nM T47768 C9UF0X 127041937 IC50 = 1250 nM T47768 C03RGT 127041938 IC50 = 11.1 nM T47768 C1OZA6 127041939 IC50 = 32 nM T47768 CZXS41 127041940 IC50 = 130.7 nM T47768 C3G9ON 127042562 Ki = 7.413 nM T47768 CP9FY0 127042605 IC50 = 66.9 nM T47768 C0XL7O 127042865 Ki = 194.98 nM T47768 C0JOS6 127042866 Ki = 2.188 nM T47768 C5G7TM 127042867 Ki = 107.15 nM T47768 CA2LP8 127042873 Ki = 263.03 nM T47768 CTZ9A0 127042874 Ki = 2041.74 nM T47768 CXMJ48 127043001 Ki = 15 nM T47768 CSV07U 127043062 Ki > 10000 nM T47768 CEGF25 127043063 Ki > 10000 nM T47768 C0CMH9 127043073 Ki > 10000 nM T47768 C3W5SX 127043074 Ki > 10000 nM T47768 CQVP14 127043075 Ki > 10000 nM T47768 C32KON 127043249 Ki > 10000 nM T47768 CZ3PC4 127043250 Ki > 10000 nM T47768 C7CKP3 127043256 Ki > 10000 nM T47768 C7XF0S 127043262 Ki > 10000 nM T47768 C6Y4NI 127043263 Ki > 10000 nM T47768 C5GU8A 127043275 Ki > 10000 nM T47768 C2Q3KT 127043276 Ki > 10000 nM T47768 CL25KU 127043277 Ki > 10000 nM T47768 CFU4H9 127043364 Ki = 9.6 nM T47768 CUX47D 127043424 Ki > 10000 nM T47768 CCP2Z8 127043425 Ki > 10000 nM T47768 C7HM0D 127043432 Ki > 10000 nM T47768 C0WM8J 127043433 Ki > 10000 nM T47768 C8CV6X 127043434 Ki > 10000 nM T47768 C30BNK 127043559 Ki = 15 nM T47768 C1GK3A 127043614 Ki > 10000 nM T47768 C61FHR 127043615 Ki > 10000 nM T47768 CCSZ68 127044528 Ki = 5 nM T47768 C4SU9L 129093829 Ki > 1000 nM T47768 C1EHU5 129188443 EC50 = 232 nM T47768 CD8FT9 129188454 Ki = 56.4 nM T47768 CC9Z0J 129188459 Ki = 604 nM T47768 CSU26Y 130431379 EC50 = 91 nM T47768 CN0BW7 130431380 EC50 = 355 nM T47768 CU8N6Z 130431382 EC50 = 48 nM T47768 C0KW2L 130431384 EC50 = 179 nM T47768 C42PDX 130431390 EC50 = 127 nM T47768 C0GEH9 130431397 EC50 = 97 nM T47768 CX4NQ9 130431408 EC50 = 224 nM T47768 CH8EK3 130431409 EC50 = 55 nM T47768 CS76FD 130431412 EC50 = 149 nM T47768 C50GOC 130442480 Ki = 9400 nM T47768 CM04RF 130442572 Ki = 4400 nM T47768 CWQO32 132584396 Ki > 10000 nM T47768 CENF10 132584397 Ki > 10000 nM T47768 CM1PN3 132584398 Ki > 10000 nM T47768 CS2H6B 132584403 Ki > 10000 nM T47768 CAVB41 132584404 Ki = 2357 nM T47768 CSK3I8 132609309 EC50 = 22.39 nM T47768 C0NUC2 132609310 EC50 = 6.607 nM T47768 C9Z6XL 132609311 EC50 = 12.59 nM T47768 CO69MW 134130798 Ki > 10000 nM T47768 CA1V9U 134131635 Ki > 10000 nM T47768 C4GPT2 134131885 Ki > 10000 nM T47768 C3Z6SV 134131949 Ki > 10000 nM T47768 C64JNH 134134355 Ki > 10000 nM T47768 C91TWF 134134844 Ki > 10000 nM T47768 C7A1PO 134137537 Ki = 1902 nM T47768 CL4K1Z 134139120 Ki > 10000 nM T47768 CK2X3O 134139232 Ki > 10000 nM T47768 C80ZPT 134139387 Ki > 10000 nM T47768 CSX32C 134141708 Ki > 10000 nM T47768 CC8V6M 134142063 Ki > 10000 nM T47768 CTQ91W 134142390 Ki > 10000 nM T47768 CG0V4O 134142896 Ki > 10000 nM T47768 CBG64F 134144504 Ki > 10000 nM T47768 CU3L0J 134145684 Ki > 10000 nM T47768 CGV52O 134147031 Ki = 1750 nM T47768 C5VAD3 134147144 Ki > 10000 nM T47768 C62SOQ 134147564 Ki > 10000 nM T47768 C8DP6W 134147710 Ki > 10000 nM T47768 CB8CI0 134147910 Ki = 892 nM T47768 CBU81N 134149168 Ki > 10000 nM T47768 C5ZD9L 134149737 Ki > 10000 nM T47768 CH97MA 134154487 Ki > 10000 nM T47768 CT2X3N 134155538 Ki = 632 nM T47768 C9QBY4 134156534 Ki > 10000 nM T47768 C13PHC 134157413 Ki > 10000 nM T47768 CLS5H3 134227139 Ki = 0.4 nM T47768 CG57MT 134563466 Ki = 71.3 nM T47768 CE5RS7 134563496 Ki > 10000 nM T47768 CAEY19 134563500 Ki = 1308 nM T47768 C82SEF 134563650 Ki = 716 nM T47768 CC3HK6 134563655 Ki = 2.4 nM T47768 C4U9EM 134563691 Ki = 504 nM T47768 CFX37T 134563695 Ki = 453 nM T47768 CPEH72 134563698 Ki = 227 nM T47768 CR74XA 134563699 Ki = 382 nM T47768 C9PN6I 134578342 Ki = 269 nM T47768 CK62WY 134578456 Ki = 306 nM T47768 CN0C9Z 134578457 Ki = 453 nM T47768 C0HNI9 134578506 Ki > 10000 nM T47768 C0JCQ2 134578518 Ki = 973 nM T47768 C1GY2T 135156251 EC50 > 10000 nM T47768 CPZ89B 135314564 Ki > 1000 nM T47768 CAX4E7 135329044 IC50 = 6400 nM T47768 CG7P3W 135329090 IC50 = 6500 nM T47768 CMS56H 135329094 IC50 = 6200 nM T47768 CUYV98 135329104 IC50 = 1200 nM T47768 CRW47P 135329122 IC50 > 10000 nM T47768 CN14XB 136036819 Ki = 25.12 nM T47768 CWE6O8 136126655 Ki = 170 nM T47768 C8IP5C 136126656 Ki = 270 nM T47768 CC6OP7 136244089 Ki > 10000 nM T47768 CQKN40 137434120 IC50 = 400 nM T47768 C0PL4B 137434175 IC50 = 110 nM T47768 CNCS34 137434196 IC50 = 1100 nM T47768 CW8LH6 137434204 IC50 = 1400 nM T47768 COQ5H7 137434366 IC50 = 1400 nM T47768 C2JK8N 137434496 IC50 = 100 nM T47768 C84KBF 137517537 EC50 = 367 nM T47768 CY93TN 137541769 EC50 = 780 nM T47768 C68GRS 137541772 EC50 = 1530 nM T47768 CX2N7C 137541775 Ki = 5.28 nM T47768 CF4UH6 137541784 Ki = 6.91 nM T47768 C2O3XI 137541786 Ki = 54.3 nM T47768 C47CEN 137541791 EC50 = 3280 nM T47768 C9PT1F 137541792 EC50 = 10000 nM T47768 C8H2LE 137541793 EC50 = 30 nM T47768 CVBP38 137541794 EC50 = 230 nM T47768 C0OKP7 137541796 EC50 = 160 nM T47768 C4R9BK 137541803 EC50 = 6600 nM T47768 C3QB8I 137541808 EC50 = 380 nM T47768 CQX9K1 137541809 EC50 = 3310 nM T47768 C07WHM 137541810 EC50 = 10 nM T47768 C3YI0Z 137541811 EC50 = 110 nM T47768 CH97XA 137541813 EC50 = 3310 nM T47768 CW6SK2 137541816 Ki = 2.27 nM T47768 C0BKU3 137631438 Ki > 10000 nM T47768 CD6OS8 137631684 EC50 = 110 nM T47768 CTH8M9 137631847 Ki = 167 nM T47768 CFT36I 137631943 Ki = 0.1 nM T47768 CB0IT4 137632188 Ki = 15.85 nM T47768 C9WUL6 137632260 Ki > 1000 nM T47768 CNC15K 137632903 Ki = 460 nM T47768 C6FEL8 137633728 Ki = 0.24 nM T47768 C4SR3G 137633741 Ki = 31.62 nM T47768 CX37GF 137633920 Ki = 0.2512 nM T47768 C7D9QE 137634365 Ki = 0.1995 nM T47768 CBW57P 137634403 Ki = 463 nM T47768 COJ2S3 137634747 Ki = 0.3981 nM T47768 CB14RN 137635022 Ki = 192 nM T47768 C8QAR1 137636327 Ki = 0.1259 nM T47768 CXB49H 137637261 EC50 > 30000 nM T47768 C5EO6T 137637552 Ki = 27.9 nM T47768 CN07MB 137637586 Ki = 0.1585 nM T47768 CUG84V 137637659 EC50 = 12100 nM T47768 C5CTQ7 137638063 Ki = 0.1585 nM T47768 COS82Q 137638460 Ki = 0.2512 nM T47768 C3NT7A 137638511 Ki = 5.04 nM T47768 C6IE4A 137638534 EC50 > 30000 nM T47768 CKR9S7 137638688 Ki = 274 nM T47768 CH4RQ3 137639037 EC50 = 904 nM T47768 C4A7CD 137639500 EC50 = 12900 nM T47768 C4CWP3 137639680 Ki = 62.8 nM T47768 CBM34G 137640362 Ki = 0.1 nM T47768 CUZ7O1 137640860 Ki = 211 nM T47768 CY2AV8 137641064 Ki = 313 nM T47768 C2OD0K 137641318 Ki > 1000 nM T47768 CMI3T0 137641479 IC50 = 144.2 nM T47768 CF7Q8M 137641618 Ki = 0.34 nM T47768 C1RAK0 137642012 Ki = 584 nM T47768 CID94R 137642522 Ki = 0.7943 nM T47768 C1IAZ5 137642772 Ki = 32.7 nM T47768 C8BZ5G 137642854 EC50 = 308 nM T47768 C4KT5V 137642888 EC50 = 3760 nM T47768 CQ9NY2 137642933 EC50 = 4870 nM T47768 CKH93R 137643506 Ki = 398 nM T47768 CAI9Z4 137643649 Ki > 10000 nM T47768 CU7MG5 137644005 Ki = 499 nM T47768 C2MRK0 137645329 Ki > 1000 nM T47768 CX7UD0 137645396 Ki = 0.1 nM T47768 CG4N0O 137646080 Ki = 17.5 nM T47768 CROM52 137646459 IC50 = 1600 nM T47768 CUHF67 137646492 EC50 = 209 nM T47768 C2OB5H 137646522 Ki = 557 nM T47768 CB34GJ 137646619 EC50 = 48.8 nM T47768 CXJ9G7 137646782 Ki = 234 nM T47768 CY1R8I 137646935 Ki = 1.585 nM T47768 C3MV2Q 137646937 Ki = 32.3 nM T47768 CTP82Z 137647554 Ki = 670 nM T47768 CY3UG7 137647869 IC50 = 2320 nM T47768 CQ76TD 137648147 Ki = 0.2512 nM T47768 CX72UG 137648224 Ki = 1.15 nM T47768 CK8EP7 137648628 Ki = 0.46 nM T47768 CH8F7A 137649449 Ki = 3.16 nM T47768 C4TDX9 137649850 Ki = 259 nM T47768 CBC86L 137650237 Ki = 0.1 nM T47768 CH84NE 137651461 EC50 = 2880 nM T47768 CZ68WR 137651510 Ki = 358 nM T47768 CCQI54 137652472 IC50 = 650 nM T47768 CV4Y7Q 137652968 Ki = 0.1 nM T47768 CK74TN 137652971 Ki = 19.9 nM T47768 C9YHQ5 137653349 Ki = 0.9 nM T47768 CS1B3U 137654001 Ki = 523 nM T47768 C6N8JM 137655206 Ki = 16.1 nM T47768 CYXW02 137655296 IC50 = 1260 nM T47768 C7P9UA 137655599 Ki = 537 nM T47768 C3KPA4 137655663 Ki = 56 nM T47768 C4D8UC 137656339 EC50 = 14200 nM T47768 CSHN48 137656887 Ki = 631 nM T47768 CY21WB 137657032 Ki = 0.455 nM T47768 CWD31I 137657725 Ki = 0.048 nM T47768 COM17P 137658558 IC50 = 794.33 nM T47768 CJZO53 137658876 IC50 = 18 nM T47768 CVU76G 137659256 EC50 > 30000 nM T47768 CM85RN 137659520 EC50 = 18300 nM T47768 C0K9SV 137659967 EC50 > 30000 nM T47768 CG8R9U 137660781 Ki = 851 nM T47768 CR0EW1 137660824 Ki = 230 nM T47768 C1XPN8 137661045 Ki = 971 nM T47768 C51IBF 137662101 EC50 = 10.23 nM T47768 CNX2Q5 137662177 Ki > 1000 nM T47768 C9LM6E 137662178 Ki = 192 nM T47768 CH6X3W 140995821 Ki = 630.96 nM T47768 CL8VT0 145946399 Ki = 1.7 nM T47768 CZ82RG 145948744 Ki = 1 nM T47768 C3EWL2 145948797 IC50 = 2.344 nM T47768 CMD58S 145948809 Ki = 6 nM T47768 C2RLY9 145948839 Ki = 0.4 nM T47768 CGA46O 145948847 Ki = 1 nM T47768 CHGW16 145948955 Ki = 27 nM T47768 C7N5LP 145948965 Ki = 4 nM T47768 CH49XK 145948968 Ki = 4 nM T47768 C5E2QA 145948981 Ki = 4 nM T47768 CI14LP 145949343 IC50 = 11300 nM T47768 CAB3N0 145950456 EC50 = 1757 nM T47768 CDA24L 145950961 Ki > 100000 nM T47768 CE9SQ4 145952136 Ki > 1000 nM T47768 CM17OA 145952209 Ki > 1000 nM T47768 CGW92C 145952721 IC50 > 30000 nM T47768 C7WT1M 145952813 IC50 = 0.016 nM T47768 C4V7GC 145952964 Ki > 1000 nM T47768 CJ89WR 145954168 EC50 > 10000 nM T47768 CVZ04C 145956193 Ki = 1080 nM T47768 C9Y8RW 145956549 Ki > 1000 nM T47768 C7SX5C 145957352 Ki > 100000 nM T47768 CFZJ34 145957574 IC50 = 79.43 nM T47768 C9X4EA 145957598 EC50 > 10000 nM T47768 C7X0LW 145958562 Ki > 100000 nM T47768 CI9XG5 145958618 Ki > 1000 nM T47768 CW2T8U 145959553 Ki > 1000 nM T47768 CY1MB9 145961131 Ki = 2.884 nM T47768 CR8WC1 145961165 Ki = 2.344 nM T47768 CIU2V6 145961844 Ki = 0.2692 nM T47768 CGR0Y1 145963106 Ki = 8.9 nM T47768 CBFE94 145963594 Ki = 2.5 nM T47768 CB6TS1 145963850 EC50 = 13 nM T47768 CO7C2S 145964378 EC50 = 75 nM T47768 CH0VD5 145964426 Ki = 2900 nM T47768 C2GNW8 145964475 EC50 = 57 nM T47768 CH78AW 145964503 EC50 = 2123 nM T47768 CM5WJ3 145964656 EC50 = 7618 nM T47768 C68KAE 145964900 EC50 > 10000 nM T47768 C1AC7N 145965538 EC50 = 111 nM T47768 C5EGT6 145965559 EC50 = 3109 nM T47768 C0IZR7 145965971 EC50 = 18 nM T47768 CY1SN2 145965998 EC50 = 1593 nM T47768 C9Q6JT 145966009 EC50 = 1403 nM T47768 CL9G3M 145966109 EC50 = 153 nM T47768 C0CTS1 145966212 EC50 = 22 nM T47768 CH06NV 145966220 EC50 = 98 nM T47768 CR34HG 145969839 Ki = 45 nM T47768 CO8B3Y 145972999 EC50 = 6423 nM T47768 C7RAE8 145973247 EC50 > 10000 nM T47768 CCL2A5 145973500 EC50 = 31 nM T47768 C64ITK 145973938 EC50 = 189 nM T47768 CS8E9V 145974224 EC50 = 373 nM T47768 CKQY21 145974323 Ki > 100000 nM T47768 C3SJK7 145974455 EC50 = 152 nM T47768 CCEU41 145974608 EC50 = 1764 nM T47768 C21ZOF 145974614 EC50 = 1354 nM T47768 C6MEK3 145975294 EC50 = 4.8 nM T47768 CQM89B 145975633 EC50 = 1236 nM T47768 CID89J 145976033 EC50 = 760 nM T47768 CG4LA1 145977533 EC50 = 148 nM T47768 CXST16 145977540 EC50 > 10000 nM T47768 CQS9N0 145978012 Ki = 48 nM T47768 C3EX4T 145978375 EC50 = 399 nM T47768 CS5Q4X 145978757 EC50 = 2975 nM T47768 C8S6LM 145978786 EC50 = 184 nM T47768 C9FVH6 145978915 Ki = 5 nM T47768 C2T1WS 145980138 Ki = 5 nM T47768 C87MSW 145980271 Ki = 10000 nM T47768 C8I7QL 145980875 Ki = 536 nM T47768 C7MK5N 145981488 Ki = 6.16 nM T47768 C63FHK 145982510 Ki = 39.3 nM T47768 C36TEU 145982515 Ki = 7.1 nM T47768 CC6A9H 145982585 Ki = 4.3 nM T47768 CU2IK5 145982792 Ki = 73.9 nM T47768 CTQV67 145982828 Ki = 485.1 nM T47768 C8MY6V 145982968 Ki = 782.9 nM T47768 CO8Z4U 145983526 Ki = 6.3 nM T47768 C4L7PT 145983969 Ki = 12.7 nM T47768 CK6F1J 145984022 Ki = 17 nM T47768 C1ONP2 145984192 Ki = 34.1 nM T47768 COP2I9 145984332 Ki = 129.5 nM T47768 C4KS7H 145984702 Ki = 303.5 nM T47768 CV41CZ 145984911 Ki = 0.037 nM T47768 CKJ5S6 145984921 Ki = 5 nM T47768 CTY73C 145984984 Ki = 7.2 nM T47768 C4N3JP 145986165 Ki = 81.1 nM T47768 CSWD95 145986663 Ki = 5 nM T47768 CNJH37 145986752 Ki = 8253 nM T47768 CUGO10 145988693 Ki = 902 nM T47768 CFOI90 145989792 Ki = 0.52 nM T47768 CO80MW 145990547 Ki = 5 nM T47768 C4L1JX 145991594 Ki = 5 nM T47768 C0FT8Y 145991902 Ki = 5.33 nM T47768 CA24SW 145991928 Ki = 7.51 nM T47768 C79MKB 145992101 EC50 = 0.28 nM T47768 CCP2U1 145992489 Ki = 328 nM T47768 CHD1X8 145994053 Ki = 5 nM T47768 C2ADQ5 145994326 EC50 = 232.5 nM T47768 C3CP1R 145994327 EC50 > 1000 nM T47768 CFO47R 145994330 EC50 > 1000 nM T47768 CBFX85 145994331 EC50 > 1000 nM T47768 CF7GX6 145994332 EC50 = 1.199 nM T47768 CL69BD 145994333 EC50 > 1000 nM T47768 CSE72Q 145994334 EC50 > 1000 nM T47768 CW6I7K 145994336 EC50 > 1000 nM T47768 C0YWU3 145994337 EC50 = 115.5 nM T47768 CVK19A 145994338 EC50 = 16.87 nM T47768 CT3MY4 145994339 EC50 = 106.4 nM T47768 C23IEG 145994341 EC50 = 158 nM T47768 CZC6W1 145994342 EC50 = 202.1 nM T47768 C9RJO2 145994343 EC50 = 15.29 nM T47768 CG9XC0 145994345 EC50 > 1000 nM T47768 CY5Q2V 146025598 EC50 = 106 nM T47768 CC2G1V 146025727 Ki = 2100 nM T47768 CKT27S 146025804 EC50 = 455.6 nM T47768 COZ7S5 146025805 EC50 = 52.41 nM T47768 CCMB45 146025806 EC50 = 203.4 nM T47768 C75JSY 146025807 EC50 = 52.41 nM T47768 C8D9PO 146167149 IC50 = 11.75 nM T47768 CUO1K6 146167150 IC50 = 5.495 nM T47768 C6P3SR 153287553 Ki > 10000 nM T47768 CV9G7Z 153287572 Ki > 10000 nM T47768 CO85KL 153287574 Ki > 10000 nM T47768 CCV4H3 153387667 IC50 = 102.33 nM T47768 CG7JL9 153387671 IC50 = 6.457 nM T47768 CXJH67 155510378 Ki = 507 nM T47768 CL6OY2 155510745 EC50 = 19.6 nM T47768 CVMK78 155512747 Ki = 19.6 nM T47768 CG95UQ 155512955 Ki = 100 nM T47768 CX4Z3F 155513383 Ki = 261 nM T47768 CI65OP 155513602 Ki = 29 nM T47768 CG4X6F 155514057 EC50 = 0.00177 nM T47768 C6F2GE 155514186 Ki = 24 nM T47768 C1UXA4 155514661 Ki = 0.23 nM T47768 CKL4N0 155515090 IC50 > 10000 nM T47768 CSM5N3 155515838 Ki = 84 nM T47768 CYRX70 155515945 Ki = 205 nM T47768 C8F9WQ 155515973 EC50 = 1900 nM T47768 CUM2N4 155515982 Ki = 2000 nM T47768 C7RT4P 155516535 Ki = 0.29 nM T47768 C3MQP5 155516545 Ki = 33 nM T47768 C3PD8O 155516811 Ki = 0.8 nM T47768 CJ80FA 155516945 IC50 > 10000 nM T47768 CAC4W6 155517219 IC50 = 70000 nM T47768 C2RPY4 155517392 EC50 > 100000 nM T47768 CYQW63 155517808 IC50 = 600 nM T47768 CUSA24 155519891 Ki > 10000 nM T47768 CWLY76 155520187 EC50 = 0.28 nM T47768 CT93LK 155520217 Ki = 105 nM T47768 CF42WX 155520785 EC50 = 1584.89 nM T47768 CB5LN9 155521072 EC50 = 0.00177 nM T47768 CY5CL2 155521553 Ki = 46.2 nM T47768 C7QCK2 155522403 EC50 = 60 nM T47768 CZ9V8E 155522689 Ki = 160 nM T47768 CWA8B7 155523094 Ki = 3.6 nM T47768 CY8XL4 155524179 Ki = 177 nM T47768 CS0LP7 155525545 Ki = 17 nM T47768 CUQC23 155525839 EC50 = 4.4 nM T47768 CSL9T1 155525842 Ki = 225 nM T47768 C24PLM 155525923 Ki > 1000 nM T47768 CDFR34 155526934 EC50 = 1.4 nM T47768 CEJI39 155527289 Ki = 166 nM T47768 C1SZ3R 155527414 IC50 = 1460 nM T47768 C5B7LS 155527564 Ki = 380 nM T47768 C7T5YS 155527675 Ki = 0.3981 nM T47768 CQV19C 155528829 Ki = 401 nM T47768 CV42PH 155529675 Ki = 40 nM T47768 CZN6H7 155529986 EC50 = 8500 nM T47768 C1FW6M 155530357 Ki = 470 nM T47768 CXH95L 155531153 Ki = 437 nM T47768 CRZ54B 155532072 Ki = 6 nM T47768 C6W5JY 155532087 Ki = 4.98 nM T47768 C3UV2R 155532761 Ki = 0.1 nM T47768 CV0UL2 155532879 Ki = 19 nM T47768 C7GU3F 155533321 Ki = 0.1585 nM T47768 CKA04B 155533331 IC50 = 0.7079 nM T47768 CTWG84 155533462 Ki = 31 nM T47768 CEG3N8 155533730 Ki = 4.1 nM T47768 CG6C1I 155535201 Ki = 137 nM T47768 C5S8MZ 155535351 Ki = 0.1 nM T47768 C05NHQ 155535754 Ki = 10000 nM T47768 CB79ZW 155536080 Ki = 1995.26 nM T47768 C2YV1C 155536562 EC50 = 3.4 nM T47768 CE6Q7N 155536593 EC50 = 17.7 nM T47768 C4RWI6 155536757 Ki = 4.8 nM T47768 CHJ59D 155537352 Ki = 7.6 nM T47768 CZT05I 155537442 Ki = 0.2512 nM T47768 CR97JX 155537513 Ki = 4.38 nM T47768 CUX51M 155538186 Ki = 76.2 nM T47768 CSZK58 155538263 Ki = 1 nM T47768 CE8UF7 155539181 IC50 = 183 nM T47768 CPDK87 155539216 Ki = 110 nM T47768 C5NE1H 155539282 Ki = 0.26 nM T47768 CX86BV 155539726 Ki = 5 nM T47768 C6IJA4 155539728 Ki = 368 nM T47768 CJF25T 155540464 Ki = 8.6 nM T47768 C0ML6F 155542107 Ki = 0.631 nM T47768 CJV8E5 155542270 Ki = 0.1259 nM T47768 C67WLH 155542684 Ki = 949 nM T47768 C85XQT 155542852 EC50 = 0.00177 nM T47768 CA27KR 155543816 IC50 = 3330 nM T47768 C27SCO 155543969 Ki = 0.1259 nM T47768 CU83VX 155544763 Ki = 80 nM T47768 CK36RG 155545176 Ki = 18.91 nM T47768 CGKR14 155546429 EC50 = 60 nM T47768 C6HGY8 155547045 Ki = 0.95 nM T47768 C4W5IM 155547169 EC50 = 52.41 nM T47768 CL36YR 155548389 Ki = 72.4 nM T47768 CY39HI 155548401 IC50 = 5754.4 nM T47768 C9VBK7 155548948 EC50 = 0.2 nM T47768 CKAN65 155549973 IC50 = 2930 nM T47768 CDFU45 155549997 EC50 < 0.51 nM T47768 C68KWY 155550260 EC50 = 0.00177 nM T47768 CFGB69 155550582 EC50 > 100000 nM T47768 C5H7AI 155551063 Ki = 0.631 nM T47768 C4S7MG 155551744 IC50 = 583 nM T47768 CX8JA1 155552185 Ki = 2300 nM T47768 C0WH2Y 155552342 Ki > 100000 nM T47768 CHSX69 155552921 Ki = 0.7943 nM T47768 C6PA3D 155553117 Ki = 96 nM T47768 CCE7J5 155553155 EC50 = 4 nM T47768 CLKV39 155554074 EC50 = 4.677 nM T47768 CHYA95 155554410 Ki = 1634 nM T47768 C81USE 155554575 Ki = 38 nM T47768 CHQ2X8 155554943 Ki = 1.4 nM T47768 CE2PJ9 155555050 EC50 = 6.2 nM T47768 CB3DO5 155556993 Ki = 240 nM T47768 CXHW52 155557070 IC50 = 71000 nM T47768 C2TD1R 155558095 IC50 = 1085000 nM T47768 CODF60 155558752 Ki = 380 nM T47768 C2Q6KU 155558968 Ki = 993 nM T47768 C7PM0A 155559194 EC50 = 0.0024 nM T47768 CF3U0D 155559400 IC50 > 2000000 nM T47768 C61BFO 155559678 Ki = 15 nM T47768 CHU9L6 155559739 Ki = 240 nM T47768 CKI47R 155560346 Ki = 0.7943 nM T47768 C20UAD 155561395 Ki > 100000 nM T47768 C8I3RS 155562884 Ki = 322 nM T47768 CJT89K 155563204 IC50 = 1500 nM T47768 CAN0G3 155563660 Ki = 406 nM T47768 C3A6ZY 155563934 Ki = 0.5 nM T47768 C4AXT9 155564059 Ki = 2.4 nM T47768 C4YJS5 155564567 EC50 = 52.41 nM T47768 CP26UB 155564632 EC50 = 1.45 nM T47768 CG5JL7 155564874 EC50 = 0.028 nM T47768 CWG3K0 155565050 Ki = 0.3162 nM T47768 CIS95O 155565113 Ki = 133 nM T47768 CEZ16B 155565184 Ki > 100000 nM T47768 CUQ25H 155566579 EC50 = 7.5 nM T47768 CL76VI 155566581 Ki = 0.48 nM T47768 CYLN53 155567284 EC50 = 0.014 nM T47768 C2MV4D 155568748 Ki = 12.59 nM T47768 CTNU54 155569410 Ki = 0.45 nM T47768 CQ0GL3 155569552 Ki = 857 nM T47768 C3N9VU 10251906 Ki = 82 nM T47768 CP9TR0 10324985 Ki > 10000 nM T47768 C6K2AI 11235101 Ki = 0.13 nM T47768 CZNV03 11495577 Ki = 1.2 nM T47768 CV52TJ 11500703 Ki = 13.5 nM T47768 CI24CL 11552110 Ki = 2.1 nM T47768 CJ23LB 11552587 Ki = 0.74 nM T47768 CS82VA 44405201 Ki = 0.13 nM T47768 C13REG 44471685 Ki = 1496 nM T47768 CFR6A5 46905974 Ki = 11 nM T47768 C3C7AZ 49796843 Ki = 1.02 nM T47768 D00FXL 44439907 Ki = 640 nM T47768 D00JPB 44434951 Ki = 0.44 nM T47768 D00NRB 6602241 Ki = 0.003 nM T47768 D00PYB 5459910 EC50 = 294 nM T47768 D00SDP 44627900 Ki = 0.08 nM T47768 D00TNR 5311081 EC50 = 0.04 nM T47768 D00XZH 44430025 Ki = 13230 nM T47768 D00YCW 44426807 Ki = 341 nM T47768 D01EPU 9804450 Ki = 0.12 nM T47768 D01HOP 44439875 Ki = 560 nM T47768 D01MUV 10314141 Ki = 3599 nM T47768 D01RFG 10086063 Ki = 0.31 nM T47768 D01SDX 44439910 Ki = 100 nM T47768 D01WMU 9820782 Ki = 2147 nM T47768 D02IMZ 44427184 Ki = 0.7 nM T47768 D02NSY 10296561 IC50 = 6700 nM T47768 D02PIG 11250396 Ki = 28 nM T47768 D02RYZ 16083055 Ki = 0.69 nM T47768 D03KAQ 44626544 Ki = 190 nM T47768 D03PTV 10022129 Ki = 377 nM T47768 D03RBD 49765077 IC50 = 721 nM T47768 D03SAV 3082718 Ki = 53 nM T47768 D03UFD 5491897 Ki = 105 nM T47768 D03UHT 44429061 Ki = 5.8 nM T47768 D03UJW 22970051 Ki = 272 nM T47768 D04FBZ 5284595 Ki = 0.19 nM T47768 D04JCJ 44434931 Ki = 643.47 nM T47768 D04JFL 16099582 Ki = 0.21 nM T47768 D04PPP 44406697 Ki = 0.16 nM T47768 D04QUB 25242485 Ki > 10000 nM T47768 D04SFK 644210 Ki > 4500 nM T47768 D04UIK 44427178 Ki = 0.11 nM T47768 D04VJE 44434061 Ki = 658.8 nM T47768 D04ZQX 44426812 Ki = 144 nM T47768 D05COL 11440685 Ki > 10000 nM T47768 D05EWZ 44444966 Ki = 14.3 nM T47768 D05EZE 10077295 EC50 = 0.1 nM T47768 D05FEQ 5359966 Ki = 0.062 nM T47768 D05JSY 10462426 Ki = 0.2 nM T47768 D05QJS 5480230 Ki = 0.94 nM T47768 D05RII 44413409 Ki = 230 nM T47768 D05XCV 44583427 Ki = 340 nM T47768 D05YXS 5462306 EC50 = 277 nM T47768 D05ZIH 45110000 Ki = 2.12 nM T47768 D05ZUX 44207909 Ki >= 1000 nM T47768 D06EES 461776 EC50 = 1.3 nM T47768 D06ESC 44577308 Ki = 12.1 nM T47768 D06IXE 11411315 Ki = 29 nM T47768 D06KFX 44583372 IC50 = 25 nM T47768 D06MQG 44430018 Ki = 2988 nM T47768 D06NST 19143 Ki = 0.16 nM T47768 D06OKE 44427174 Ki = 1.4 nM T47768 D06PHT 10269001 Ki = 207 nM T47768 D06PVO 44426806 Ki = 2298 nM T47768 D06QGJ 52946209 IC50 > 30000 nM T47768 D06SZI 44429060 Ki = 160 nM T47768 D06YMS 6917707 EC50 = 128.82 nM T47768 D07BPA 11645313 Ki > 10000 nM T47768 D07CIU 9924923 Ki = 940 nM T47768 D07DFD 44427176 Ki = 5.3 nM T47768 D07FCB 9925737 Ki = 6265 nM T47768 D07HFU 44429064 Ki = 12 nM T47768 D07ICW 11556976 Ki = 20 nM T47768 D07JIQ 44439882 Ki = 1200 nM T47768 D07KTF 24873526 Ki = 41 nM T47768 D07NMH 10093682 Ki = 1057 nM T47768 D07PPK 44406272 Ki > 465 nM T47768 D07QUY 44583388 Ki = 43 nM T47768 D08DVV 44430026 Ki = 8899 nM T47768 D08IWF 44427180 Ki = 1.2 nM T47768 D08LIT 11641503 EC50 = 5.17 nM T47768 D08NJB 16733487 EC50 = 2.65 nM T47768 D08QBS 44178080 IC50 > 10000 nM T47768 D08QBU 44430029 Ki = 3364 nM T47768 D08RPH 11255361 Ki = 3.7 nM T47768 D08SCK 11664525 Ki = 0.46 nM T47768 D08TFY 10043439 Ki = 407 nM T47768 D09BWX 44583373 IC50 = 21 nM T47768 D09BYD 20481138 Ki = 74 nM T47768 D09DUE 44429063 Ki = 3.2 nM T47768 D09FJY 9863568 Ki = 246 nM T47768 D09FLC 44627904 Ki = 0.34 nM T47768 D09GQP 15384271 IC50 = 894 nM T47768 D09GSD 11721803 Ki = 19.9 nM T47768 D09KBQ 131534 Ki = 0.11 nM T47768 D09LRO 44430008 Ki = 705 nM T47768 D09RPR 16737207 Ki > 10000 nM T47768 D09RUY 44627790 Ki = 0.26 nM T47768 D09SBU 44583393 Ki = 22 nM T47768 D09TCT 44577349 Ki = 112.5 nM T47768 D09UKS 11303119 Ki = 7.1 nM T47768 D09VRT 44426814 Ki = 24 nM T47768 D0A0GU 44247568 Ki > 10000 nM T47768 D0A3YH 24853671 EC50 = 3.28 nM T47768 D0A5MU 44390358 Ki = 3.5 nM T47768 D0A9AJ 44439901 Ki = 1100 nM T47768 D0AC0A 10047612 Ki = 58 nM T47768 D0B8MY 9897164 Ki = 0.09 nM T47768 D0BI4T 53315878 Ki > 10000 nM T47768 D0C2UQ 44427183 Ki = 0.12 nM T47768 D0C7MP 44429062 Ki = 1.4 nM T47768 D0D0UP 10315818 Ki = 1734 nM T47768 D0D1VB 11498201 Ki > 1000 nM T47768 D0D5QV 9838803 Ki = 8.6 nM T47768 D0D5VD 44583375 Ki = 120 nM T47768 D0D8AN 13374610 Ki = 0.24 nM T47768 D0D9BB 10427620 Ki = 11540 nM T47768 D0E0TD 44434950 Ki = 0.15 nM T47768 D0E6GH 44565511 Ki = 0.34 nM T47768 D0E6IT 44439879 Ki > 10000 nM T47768 D0ED2I 11016572 Ki = 0.16 nM T47768 D0F1EB 44417373 Ki = 0.46 nM T47768 D0F4AN 44427182 Ki = 3.7 nM T47768 D0F8AX 44430024 Ki = 18365 nM T47768 D0F8CD 45487600 Ki = 8.67 nM T47768 D0F8CV 5462471 Ki = 0.28 nM T47768 D0FF6S 16038374 IC50 = 10000 nM T47768 D0G1IF 9576413 Ki = 1.445 nM T47768 D0G4FA 10384734 Ki = 11050 nM T47768 D0G4NM 104787 IC50 = 1.6 nM T47768 D0G7DF 44426827 Ki = 147 nM T47768 D0G7FB 9798655 Ki = 1.5 nM T47768 D0H0KP 44434946 Ki = 22.26 nM T47768 D0H1BU 10864183 Ki = 0.16 nM T47768 D0H2CI 44456192 Ki = 390 nM T47768 D0HB6O 44439880 Ki = 9.8 nM T47768 D0HN2M 44430609 Ki = 74.13 nM T47768 D0I1NG 44434058 Ki = 0.07 nM T47768 D0I1ZN 44583428 Ki = 360 nM T47768 D0I2CE 44583376 Ki = 37 nM T47768 D0IL9H 44430013 Ki = 11430 nM T47768 D0IQ0S 45487602 Ki = 122 nM T47768 D0IU2K 44577307 Ki = 705 nM T47768 D0IY2V 44429065 Ki = 22 nM T47768 D0J3NK 44427177 Ki = 0.29 nM T47768 D0J5IR 44555371 Ki = 4.97 nM T47768 D0J5JO 44430009 Ki = 273 nM T47768 D0J7VL 44439873 Ki > 10000 nM T47768 D0JH5D 44430007 Ki = 589 nM T47768 D0JX3P 44577306 Ki = 3190 nM T47768 D0K0OT 1329 Ki > 100000 nM T47768 D0K1BV 44628003 Ki = 11 nM T47768 D0K4XQ 44427175 Ki = 4.8 nM T47768 D0KQ8A 44555370 Ki = 2.32 nM T47768 D0L2CT 24768355 Ki = 9.5 nM T47768 D0L5DN 11392313 Ki = 1.3 nM T47768 D0L5MW 181743 Ki = 7265 nM T47768 D0L6QN 10070040 Ki = 0.14 nM T47768 D0L8LX 123704 Ki = 12 nM T47768 D0L8YY 10066285 Ki = 5.24 nM T47768 D0L9YP 44254503 Ki = 2700 nM T47768 D0M1YV 16747727 Ki = 18000 nM T47768 D0N3GU 44577305 Ki = 72.7 nM T47768 D0NA7G 16083058 Ki = 1100 nM T47768 D0NE3U 5485199 Ki = 1.585 nM T47768 D0O1JD 44434057 Ki = 2.25 nM T47768 D0O2LD 5324289 EC50 = 5600 nM T47768 D0O6SB 443408 Ki = 0.07 nM T47768 D0O7JV 44426810 Ki = 37 nM T47768 D0OH7D 5310988 Ki = 10.5 nM T47768 D0P2DF 15747210 Ki = 37.3 nM T47768 D0P2TT 73354725 Ki > 10000 nM T47768 D0P3FP 44426808 Ki = 29 nM T47768 D0P5IH 44583387 Ki = 170 nM T47768 D0P5QI 44626540 Ki = 15 nM T47768 D0P6FF 44627901 Ki = 1.7 nM T47768 D0P8TI 11466688 Ki > 10000 nM T47768 D0PN3P 44439877 Ki = 1200 nM T47768 D0Q5AJ 44365804 Ki = 66 nM T47768 D0Q6CF 44583374 Ki = 670 nM T47768 D0Q9TQ 10043898 Ki = 412 nM T47768 D0QH4A 10089987 Ki = 771 nM T47768 D0R0OZ 119303 Ki = 150 nM T47768 D0R2VL 44434060 Ki = 1008 nM T47768 D0R4QF 11431898 Ki = 12 nM T47768 D0R5TA 5311080 EC50 = 0.001 nM T47768 D0R6VF 6540640 Ki = 0.25 nM T47768 D0R6VX 45487601 Ki = 56.23 nM T47768 D0R7LY 16733485 EC50 = 2.35 nM T47768 D0R9AP 44439872 Ki = 1400 nM T47768 D0S2OA 10388166 Ki = 21455 nM T47768 D0S3TZ 5748293 Ki = 10.6 nM T47768 D0S5BJ 5459823 EC50 = 28 nM T47768 D0S5FN 44439876 Ki = 9.8 nM T47768 D0SC3W 44406704 Ki = 14 nM T47768 D0SE9S 9887077 Ki = 65 nM T47768 D0T2RY 9948320 Ki >= 1000 nM T47768 D0T4ZY 44426817 Ki = 451 nM T47768 D0T6OQ 10021946 Ki = 0.71 nM T47768 D0T9KE 44430016 Ki = 983 nM T47768 D0U3UM 13493 Ki = 0.2 nM T47768 D0U5OP 11580459 Ki = 1000 nM T47768 D0U7JS 44439866 Ki = 18 nM T47768 D0U7PT 25075996 EC50 = 213.8 nM T47768 D0UG5M 9956146 Ki = 0.96 nM T47768 D0UR7D 44390359 Ki = 0.5 nM T47768 D0V3OY 105104 IC50 = 250 nM T47768 D0VO7C 10677974 Ki = 5.62 nM T47768 D0W0CO 44627903 Ki = 1.7 nM T47768 D0W1YD 44439896 Ki > 10000 nM T47768 D0W2DN 44427179 Ki = 0.3 nM T47768 D0W3PR 44555372 Ki = 4.56 nM T47768 D0W3VT 10091033 Ki = 936 nM T47768 D0WT7H 5311018 Ki = 0.41 nM T47768 D0X4SX 10317947 Ki = 1649 nM T47768 D0X5TB 44439905 Ki = 19 nM T47768 D0X7LC 11061906 Ki = 610 nM T47768 D0XX1Y 44426828 Ki = 3728 nM T47768 D0Y2HI 11635818 Ki = 1.48 nM T47768 D0Y5LJ 10336926 Ki = 4554 nM T47768 D0Y5ZP 44626534 Ki = 17 nM T47768 D0Y7CI 123924 EC50 = 0.14 nM T47768 D0Y7KE 44430012 Ki = 3433 nM T47768 D0Y8NO 22977851 Ki = 3.1 nM T47768 D0Y9RD 44428865 Ki = 225.9 nM T47768 D0YU5H 44434949 Ki = 2.43 nM T47768 D0Z5JD 9985128 Ki = 11.4 nM T47768 D0Z8JX 44583386 Ki = 40 nM T47768 D0ZE2W 44430028 Ki = 10390 nM T06770 C26SVD 451777 IC50 = 250000 nM T06770 C5ZJQ3 488950 IC50 = 30000 nM T06770 C7GFT4 488962 IC50 > 100000 nM T06770 C8Q9JO 16134139 IC50 = 0.86 nM T06770 C7EC9G 16134140 IC50 = 0.84 nM T06770 C3A0YM 16134186 IC50 = 0.34 nM T06770 C6JQ3C 16143364 IC50 = 0.35 nM T06770 C6PG2R 46186917 IC50 = 9600 nM T06770 C9HL2I 46200686 IC50 = 9300 nM T06770 CRC8H5 53324414 IC50 = 83200 nM T06770 CG64CF 71596849 IC50 = 2.18 nM T06770 CZ7R4M 71597777 IC50 = 2.27 nM T06770 C8ML9U 122184656 IC50 = 17.74 nM T06770 C0FJ8S 122184657 IC50 = 17.7 nM T06770 CZ1R0G 122184658 IC50 > 2250 nM T06770 CF5P4J 122184659 IC50 = 58.79 nM T06770 D03QJA 11718722 IC50 = 1.71 nM T33489 D00ZFP 5870 IC50 = 51000 nM T33489 D08QMX 5757 IC50 = 84000 nM T33489 D04ZND 6918339 IC50 = 16 nM T33489 D07ZNI 9804302 IC50 = 39 nM T33489 D0D3PF 6918191 IC50 > 10000 nM T33489 CJ7AG2 66413 IC50 = 19600 nM T33489 C57CIN 66428 IC50 = 14400 nM T33489 CKFQ24 74626 IC50 > 30000 nM T33489 C2BPM9 92846 IC50 > 50000 nM T33489 CE10GB 233494 IC50 = 2800 nM T33489 CLI5U8 233496 IC50 = 17000 nM T33489 C16WHM 233497 Ki = 1400 nM T33489 CTWQ60 233498 IC50 = 26000 nM T33489 CS7IK6 248293 IC50 = 293 nM T33489 C5IQZ0 460028 IC50 = 41000 nM T33489 CP9L7I 3052707 IC50 = 750000 nM T33489 C3T1JC 3081351 IC50 = 55.8 nM T33489 CJ1U7P 4369413 IC50 = 277 nM T33489 CK17YZ 4369414 IC50 = 39 nM T33489 C5K7RG 6871072 IC50 > 100000 nM T33489 CHJ85P 6904461 IC50 = 24000 nM T33489 CO8PK2 6904720 IC50 = 4000 nM T33489 C13SAQ 6913081 Ki = 15000 nM T33489 CCTL65 9747438 IC50 > 100000 nM T33489 CVB91A 9763740 IC50 = 13000 nM T33489 CU54PO 9800523 IC50 = 37 nM T33489 CFDU43 9804585 Ki = 35900 nM T33489 CGB13M 9813380 IC50 = 31600 nM T33489 CHUQ47 9819457 IC50 = 1620 nM T33489 CTXR52 9820272 IC50 = 0.15 nM T33489 C4VK7F 9822055 IC50 = 78 nM T33489 CA7CJ6 9838699 IC50 = 722 nM T33489 C8EJ2Y 9842908 IC50 = 16 nM T33489 CQ6X1B 9844582 IC50 = 55.8 nM T33489 CY86ZM 9847757 IC50 = 0.81 nM T33489 CR3JH7 9864415 IC50 = 5.6 nM T33489 CY94DX 9883122 IC50 = 134 nM T33489 CV4B3K 9885452 IC50 = 8700 nM T33489 C6Q1WE 9888338 IC50 = 11 nM T33489 CF1ZH7 9905590 IC50 = 1620 nM T33489 CMVA90 9912519 IC50 = 1 nM T33489 CSN58Y 9913185 IC50 = 30 nM T33489 CV1HT9 9926309 IC50 = 3400 nM T33489 C2CSZ8 9926833 IC50 = 5.6 nM T33489 C6MBI0 9926837 IC50 = 3400 nM T33489 CH52KG 9927771 IC50 = 45 nM T33489 C07OEN 9931239 IC50 = 45 nM T33489 C4HQT0 9938946 IC50 = 160 nM T33489 CI8FG5 9949110 IC50 = 62 nM T33489 C61TJX 9950057 IC50 = 190 nM T33489 C14POL 9951107 IC50 = 0.62 nM T33489 CE6VK2 9952001 IC50 = 0.44 nM T33489 C3JT1B 9952398 IC50 = 0.34 nM T33489 CZ98XG 9976564 IC50 = 1020 nM T33489 CJ9K1V 9981999 Ki > 500000 nM T33489 CXD28H 10015065 IC50 = 912000 nM T33489 CG73UY 10023547 IC50 = 70 nM T33489 CU5Y2K 10039578 IC50 = 5000 nM T33489 C1XBV4 10059221 IC50 = 120000 nM T33489 COI6Y1 10059630 IC50 = 1000 nM T33489 CB75IJ 10093657 IC50 = 370 nM T33489 CRN29P 10104483 IC50 = 1585000 nM T33489 C5I3VO 10108748 IC50 = 120000 nM T33489 CEG43I 10113372 IC50 = 0.11 nM T33489 CRP4I5 10158995 IC50 = 1 nM T33489 C4JSN9 10159931 IC50 = 74 nM T33489 CMK8V0 10178623 IC50 = 12 nM T33489 CYWB12 10179510 IC50 = 52 nM T33489 C4WC7S 10198111 IC50 = 254000 nM T33489 C2VW0S 10198275 IC50 = 3400 nM T33489 COF37J 10224895 IC50 = 1 nM T33489 CF8QZ0 10226631 IC50 = 1 nM T33489 CNOA18 10226998 IC50 = 1 nM T33489 CN7C9F 10229969 IC50 = 23 nM T33489 CPI7V8 10273661 IC50 = 1 nM T33489 CKBA97 10297551 IC50 = 1 nM T33489 CLM67K 10323549 Ki = 530 nM T33489 C9KJ0F 10333280 IC50 = 30 nM T33489 CER52W 10334856 IC50 = 420 nM T33489 C5YOW4 10360393 Ki = 140000 nM T33489 CC0L2U 10360590 IC50 = 1 nM T33489 C3ZNC9 10363059 IC50 = 236 nM T33489 CY62IF 10393107 Ki = 76 nM T33489 COX16G 10420257 IC50 = 190500 nM T33489 C5IK7H 10420920 IC50 = 330000 nM T33489 CXZ93W 10498888 IC50 = 62 nM T33489 C0HAU9 10500968 IC50 = 110 nM T33489 C74OUY 10538931 IC50 = 380 nM T33489 CM1C0Y 10546207 IC50 = 930 nM T33489 CSD0G7 10568309 IC50 = 3490 nM T33489 CX0L3C 10595371 IC50 = 780 nM T33489 CY9A4V 10596211 IC50 = 440 nM T33489 CE86YZ 10598136 IC50 = 12 nM T33489 C9QXE8 10598137 IC50 = 25 nM T33489 CSE7C8 10599292 IC50 = 0.39 nM T33489 CS04NU 10621641 IC50 = 520 nM T33489 CT2N5H 10625121 IC50 = 0.15 nM T33489 CIL6K2 10643278 IC50 = 620 nM T33489 CRW3I1 10646335 IC50 = 640 nM T33489 C6Y9MK 10668254 IC50 = 110 nM T33489 CF5O3L 10669382 IC50 = 120 nM T33489 CCH15B 10693977 IC50 = 80 nM T33489 CF9U4R 10713699 Ki = 250 nM T33489 COM63V 10717985 IC50 = 24 nM T33489 CY0D5B 10736103 IC50 = 1980 nM T33489 C67YPW 10739143 Ki = 57000 nM T33489 C9P5NL 10741814 IC50 = 840 nM T33489 C8QCG4 10742925 IC50 = 22 nM T33489 CKQ7G9 10751772 IC50 = 1380 nM T33489 CCYQ17 10762347 IC50 = 130 nM T33489 C0QDH7 10765585 IC50 ~ 6000 nM T33489 CV9I4K 10811643 IC50 ~ 1000 nM T33489 C0WG5F 10871017 IC50 = 6330 nM T33489 CY7PA2 10872022 IC50 = 22400 nM T33489 CM5B1D 10883602 IC50 = 40 nM T33489 C5XT9Q 10914912 IC50 = 5640 nM T33489 CO01VY 10925217 IC50 = 2580 nM T33489 C71EUA 10925409 IC50 = 280 nM T33489 CFR37G 10957163 IC50 = 3300 nM T33489 CW78XH 10958393 IC50 = 24300 nM T33489 CZP94Y 11023743 IC50 = 50 nM T33489 CWR14N 11079165 IC50 = 5133 nM T33489 CV6UL9 11087274 IC50 > 100000 nM T33489 COXR05 11099671 IC50 = 62 nM T33489 CQ1K9W 11111671 IC50 = 291 nM T33489 CLP52V 11128562 IC50 = 31600 nM T33489 C7QPX9 11163126 IC50 > 180 nM T33489 CWKT25 11163616 IC50 = 180 nM T33489 CZ75AJ 11164808 IC50 = 1800 nM T33489 CEF2M0 11185919 IC50 > 530 nM T33489 CE6UZ1 11187275 IC50 > 530 nM T33489 C2CHY5 11188898 IC50 = 130 nM T33489 COK36N 11198029 IC50 = 180 nM T33489 CU0QH3 11211176 IC50 = 1000 nM T33489 C7H1AO 11246448 IC50 = 44 nM T33489 CS41OQ 11372800 IC50 = 890 nM T33489 CV4G9S 11384786 IC50 = 10 nM T33489 CI47OG 11416049 IC50 > 180 nM T33489 C2NVZ4 11461061 IC50 > 530 nM T33489 CVM9Z5 11461877 IC50 > 180 nM T33489 CKX82N 11473200 IC50 > 180 nM T33489 C6UM4W 11473201 IC50 > 180 nM T33489 CEFC74 11495013 IC50 > 10000 nM T33489 C3DG9A 11519258 Ki = 12 nM T33489 CV3U7F 11530377 IC50 = 40000 nM T33489 CD42HQ 11539191 IC50 = 1200 nM T33489 CHJB42 11567631 IC50 > 10000 nM T33489 CF51ZE 11568594 IC50 > 10000 nM T33489 COX19Z 11581191 IC50 = 140 nM T33489 CCB82K 11596108 Ki = 28000 nM T33489 CKTA53 11603462 IC50 = 590 nM T33489 CM8P2L 11609292 IC50 = 8 nM T33489 C9QOK8 11654142 IC50 > 10000 nM T33489 C4VZO5 11709992 Ki = 350000 nM T33489 C0MD6A 11732219 IC50 = 20 nM T33489 C59ANU 11758921 IC50 = 672 nM T33489 CY58WN 11781904 IC50 = 11200 nM T33489 CS89RK 11782082 IC50 = 437 nM T33489 CT3HQ9 11808626 IC50 = 0.047 nM T33489 C2MQ5U 11824989 IC50 = 140 nM T33489 C34KXP 12020775 IC50 = 3820 nM T33489 C18LXJ 12411101 IC50 > 10000000 nM T33489 C2TL6I 14334327 Ki = 1500 nM T33489 C05GMJ 15081867 IC50 = 4800 nM T33489 CK3CB6 15941002 IC50 = 200 nM T33489 C0N6GZ 15941003 IC50 = 70 nM T33489 C0DE3Y 15941004 IC50 = 1 nM T33489 C9UP0N 15941005 IC50 = 2.4 nM T33489 C31YEX 15949288 IC50 > 10000 nM T33489 CNU47L 16098586 IC50 = 190 nM T33489 CBL30A 16126879 IC50 = 160 nM T33489 CCB2Z6 16730515 IC50 = 3 nM T33489 C0E5GW 16748375 IC50 = 1300 nM T33489 C2RWY0 16748502 IC50 > 100000 nM T33489 CCX08Z 16748503 IC50 > 100000 nM T33489 CHT81I 16748506 IC50 > 100000 nM T33489 CU72RY 16748507 IC50 = 810 nM T33489 CM8D5C 16748612 IC50 > 100000 nM T33489 C3CHP0 16748613 IC50 = 43000 nM T33489 C95KCA 16748614 IC50 = 13000 nM T33489 CH6G0F 16748615 IC50 = 60000 nM T33489 CGK7C5 16748616 IC50 = 58000 nM T33489 CAHQ89 16748618 IC50 = 20000 nM T33489 CW1S9H 16748719 IC50 = 4000 nM T33489 CW7A6P 16748720 IC50 = 4200 nM T33489 C2X5QM 16748721 IC50 > 100000 nM T33489 C25HVZ 16748722 IC50 = 730 nM T33489 C1AZ4X 16748723 IC50 > 100000 nM T33489 CG51DU 16748724 IC50 = 2500 nM T33489 CH26RQ 16748725 IC50 = 35000 nM T33489 C14OZA 16748726 IC50 = 20000 nM T33489 CFX0I7 16749017 IC50 = 190 nM T33489 CEB09A 16749022 IC50 > 10000 nM T33489 CBU08D 16749337 IC50 = 380 nM T33489 C6U7AF 16749441 IC50 = 536 nM T33489 CYG64Q 17756307 IC50 = 520 nM T33489 C5OIL2 17756517 IC50 = 40 nM T33489 C8EF7J 19108716 IC50 = 537000 nM T33489 CSKO15 21044501 IC50 > 10000 nM T33489 CVA07N 21044507 IC50 = 1000 nM T33489 CN31XE 21925106 IC50 = 1024 nM T33489 CWBS90 21925109 IC50 = 0.4 nM T33489 CK2ZS8 21976856 IC50 = 476 nM T33489 CHW5O3 23585518 IC50 = 5500 nM T33489 CN84RU 23661503 IC50 = 215000 nM T33489 CSQ93A 23718123 IC50 = 4000 nM T33489 CFH3B4 24202898 IC50 = 100 nM T33489 C3ADE6 24807254 IC50 = 1400 nM T33489 CY27CS 24901646 IC50 = 920 nM T33489 CD9IV7 24901647 IC50 = 2600 nM T33489 CMFU23 24901648 IC50 = 4633 nM T33489 CTJ76G 24901649 IC50 = 553 nM T33489 CON29S 25141424 IC50 = 1200 nM T33489 CW5F9D 44267234 IC50 = 1380 nM T33489 CPT05F 44277007 IC50 = 80000 nM T33489 C8NCR1 44318681 IC50 = 3400 nM T33489 CF3A0B 44318828 IC50 = 3400 nM T33489 C4ZF1C 44318829 IC50 = 3400 nM T33489 CB13OM 44318896 IC50 = 39800 nM T33489 CV53SO 44319150 IC50 = 3400 nM T33489 CVU95M 44347238 Ki = 5800 nM T33489 CFCE82 44347239 IC50 = 13000 nM T33489 C2NXY6 44347254 Ki = 1850 nM T33489 C61RZF 44347261 IC50 > 30000 nM T33489 CX38KL 44347262 IC50 = 4320 nM T33489 CHV5Q7 44347439 IC50 > 100000 nM T33489 C5S9NO 44347499 IC50 = 37100 nM T33489 C7G8KH 44347507 IC50 = 910 nM T33489 CM93NI 44347508 IC50 = 39200 nM T33489 C89UPY 44357150 IC50 = 5.6 nM T33489 CCXJ45 44357408 IC50 = 11 nM T33489 C1R4WT 44364826 IC50 = 11 nM T33489 C3EA1Q 44389144 IC50 > 100000 nM T33489 C37TPW 44389145 IC50 > 100000 nM T33489 C1JZ7K 44389160 IC50 = 2800 nM T33489 CACX67 44389161 IC50 = 1900 nM T33489 C4EH1Z 44389163 IC50 = 3600 nM T33489 CVY7L4 44389164 IC50 = 8600 nM T33489 CYZ2R3 44389185 IC50 = 210 nM T33489 C1WO8L 44389189 IC50 > 100000 nM T33489 CYQ2Z4 44389190 IC50 = 1790 nM T33489 CB9NC2 44389195 IC50 = 71000 nM T33489 C6VI4A 44389204 IC50 = 10200 nM T33489 C80KEG 44389214 IC50 = 6100 nM T33489 CGUN50 44389219 IC50 = 450 nM T33489 CSY7H5 44394154 IC50 > 10000 nM T33489 C0C3QP 44394171 IC50 = 1500 nM T33489 CE5S8W 44398941 IC50 > 10000 nM T33489 COW9E0 44459222 IC50 = 2089000 nM T33489 C4VS7T 44459223 IC50 = 537000 nM T33489 CX6NK9 44459233 IC50 = 257000 nM T33489 CVJZ75 44459343 IC50 = 2089000 nM T33489 C8P4EB 44459430 IC50 = 300000 nM T33489 CNW10Y 44459431 IC50 = 560000 nM T33489 C92QWL 44521066 IC50 = 5.5 nM T33489 CVO41F 45140953 IC50 = 35 nM T33489 CRZ6N5 45140954 IC50 > 10000 nM T33489 C01WQZ 45141152 IC50 > 10000 nM T33489 CC3FT1 45141154 IC50 > 10000 nM T33489 CMTB56 45141155 IC50 > 10000 nM T33489 C8PB0I 45141156 IC50 = 32.6 nM T33489 CCIP58 45141367 IC50 > 10000 nM T33489 C2YJ8N 45141369 IC50 = 6333 nM T33489 C5CB0P 45141371 IC50 = 28.6 nM T33489 CGK5O7 45141601 IC50 = 29 nM T33489 C0C3AW 45141603 IC50 > 10000 nM T33489 C8QCH2 49779539 IC50 = 26 nM T33489 C7V2XL 49779540 IC50 = 205 nM T33489 CX5LZ9 50915159 IC50 = 0.13 nM T33489 C8N5OK 50991893 IC50 = 17 nM T33489 C1VF4Z 51346982 IC50 = 0.83 nM T33489 C6Y3EL 51346989 IC50 = 22 nM T33489 CBG60L 52918369 IC50 = 199 nM T33489 CGW6J8 53317154 IC50 = 43000 nM T33489 CF5J2O 53318064 IC50 > 50000 nM T33489 CF0YL2 53318824 IC50 > 50000 nM T33489 CQ9U3H 53320271 IC50 > 50000 nM T33489 C9OPT6 53320278 IC50 = 240 nM T33489 CCNP36 53321604 IC50 = 55 nM T33489 CRL4C0 53322427 IC50 > 50000 nM T33489 CKIB45 53322482 Ki = 72700 nM T33489 CUW47A 53325061 IC50 = 120 nM T33489 CA32FG 53325544 IC50 = 2900 nM T33489 C3CP6T 53326333 IC50 > 50000 nM T33489 COQ76B 53326448 IC50 > 50000 nM T33489 CN0SW9 53326827 IC50 = 2900 nM T33489 CSQ45A 53326828 IC50 = 2.3 nM T33489 CG78PF 54769379 IC50 = 126 nM T33489 C8US4R 56658390 Ki = 30 nM T33489 CJP8L2 56658391 IC50 = 224000 nM T33489 CA26QE 56658532 IC50 = 145000 nM T33489 C69JCY 56670232 Ki = 85 nM T33489 CZS90G 56675651 IC50 = 6700 nM T33489 CA3G2I 57390742 IC50 = 341 nM T33489 C6XWH8 57390743 IC50 = 364 nM T33489 C16FWY 57390744 IC50 = 207 nM T33489 CKPO26 57390745 IC50 = 26 nM T33489 CD6C1G 57390788 IC50 = 18 nM T33489 C9MH5Z 57390789 IC50 = 9 nM T33489 CV8GZ5 57391604 IC50 = 479 nM T33489 CI2C5B 57391605 IC50 = 73 nM T33489 CW45PE 57392552 IC50 = 51 nM T33489 CBS2K4 57392600 IC50 = 39 nM T33489 CW2NF9 57392601 IC50 = 67 nM T33489 CT78RD 57392602 IC50 = 137 nM T33489 C0WPZ5 57393356 IC50 = 112 nM T33489 C8CW7A 57394276 IC50 = 261 nM T33489 C5S1YG 57394319 Ki = 23 nM T33489 C5PC2G 57394320 IC50 = 190 nM T33489 CE7WA2 57396903 IC50 = 749 nM T33489 CHV63P 57397829 IC50 = 44 nM T33489 C4OWV5 57397893 IC50 = 20 nM T33489 CRG9S1 57398652 IC50 = 74 nM T33489 C8TI0H 57399535 IC50 = 493 nM T33489 CUL12P 57399536 IC50 = 271 nM T33489 C4TG1A 57399537 IC50 = 90 nM T33489 CY98JM 57400268 IC50 = 65 nM T33489 CO80SY 57400333 IC50 = 193 nM T33489 C9DKM0 57400334 IC50 = 35 nM T33489 C34UFT 57401256 IC50 = 343 nM T33489 C9OY1C 57403047 IC50 = 62 nM T33489 C63ASE 57403822 IC50 = 23 nM T33489 C97FZU 68561433 IC50 = 367 nM T33489 CFK2H7 70680992 IC50 = 0.8 nM T33489 CRH97S 70680993 IC50 > 10000 nM T33489 C4KFB1 70680994 IC50 > 10000 nM T33489 C3U5TS 70680995 IC50 > 10000 nM T33489 C6LG9Q 70683120 IC50 > 10000 nM T33489 C9U0KZ 70687355 IC50 > 10000 nM T33489 C67EAZ 70689407 IC50 = 0.1 nM T33489 C8TJ0R 70691515 IC50 = 1.2 nM T33489 C0UC3D 70695719 IC50 > 10000 nM T33489 CHC8L4 71614085 IC50 = 2.5 nM T33489 C84HSR 77460992 IC50 = 3.9 nM T33489 CT72IX 86302456 IC50 = 170 nM T33489 CEO8A1 86303760 IC50 = 8 nM T33489 C83TNX 90654353 IC50 = 88 nM T33489 C6PU7E 90659767 IC50 = 8.9 nM T33489 CJZ29C 90661603 IC50 = 15000000 nM T33489 C79CYB 100986474 IC50 = 72 nM T33489 CJSF86 101129698 IC50 = 13 nM T33489 CZP9M7 101129699 IC50 = 60 nM T33489 C2K4DX 101129700 IC50 = 75 nM T33489 CF13NO 118718106 Ki = 16000 nM T33489 CXY8Z0 121468992 IC50 = 16.6 nM T33489 C7KTD1 122184378 IC50 = 12 nM T33489 CG58QW 122184379 IC50 = 11 nM T33489 CV8Y6A 122184380 IC50 = 8 nM T33489 C5BU9A 122184381 Ki = 1 nM T33489 C3AD4Z 122184382 IC50 = 50 nM T33489 C0QA8I 122184383 IC50 = 67 nM T33489 C43OBR 122184384 IC50 = 81 nM T33489 C80PMZ 122184385 IC50 = 33 nM T33489 CGPZ20 122184386 IC50 = 49 nM T33489 C82GOQ 122184387 IC50 = 95 nM T33489 C70LXO 122184388 Ki = 2.5 nM T33489 C01CWK 122184987 IC50 = 94 nM T33489 CM5A7F 122184989 IC50 = 66 nM T33489 CWM21G 122184994 IC50 = 139 nM T33489 CXD58W 122188102 IC50 = 33780 nM T33489 C4XYZ5 122188103 IC50 = 7760 nM T33489 CB0LR7 122188104 IC50 = 7040 nM T33489 C4Q8SF 122188105 IC50 = 75020 nM T33489 CNP7D3 122188106 IC50 = 14830 nM T33489 C0FC7Q 122188107 IC50 = 6770 nM T33489 C58YBA 122188108 IC50 = 26940 nM T33489 C8N6LZ 122188145 IC50 = 860 nM T33489 CKRA78 122188146 IC50 = 5510 nM T33489 CU6X7D 122188147 IC50 = 74330 nM T33489 CQ43IS 122188148 IC50 = 109970 nM T33489 C49FPZ 122188149 IC50 = 88830 nM T33489 CPQ2V0 122188150 IC50 = 1010 nM T33489 C6AK5G 122191559 IC50 = 1 nM T33489 C9YBR2 122191560 IC50 = 1 nM T33489 CO7E3N 122191580 IC50 = 3100 nM T33489 C03SBU 122191587 IC50 = 3000 nM T33489 C0WI6K 122191772 IC50 > 10000 nM T33489 CGJU04 122191773 IC50 = 300 nM T33489 CZ7IL5 122215949 Ki = 2800 nM T33489 C54CSV 127043133 IC50 = 1 nM T33489 CK5YO8 127046605 IC50 = 1.7 nM T33489 C03MCP 127048196 IC50 = 30 nM T33489 C8DIC5 127048358 IC50 = 470 nM T33489 CJ3SV8 127048543 IC50 = 30 nM T33489 CI73MW 127048544 IC50 = 30 nM T33489 CUTF91 127048723 IC50 = 310 nM T33489 CO5DB8 127049050 IC50 = 190 nM T33489 CFP6H3 127049051 IC50 = 240 nM T33489 CML07N 127049232 IC50 = 0.05 nM T33489 CAB18N 127049525 IC50 = 44 nM T33489 CFA2P3 127049526 IC50 = 44 nM T33489 CGCZ03 127049548 IC50 = 0.04 nM T33489 C7WFA6 127049549 IC50 = 21 nM T33489 C29WMP 127049550 Ki = 250 nM T33489 CMA38E 127049551 Ki = 82000 nM T33489 C7LXE5 127050162 IC50 = 44 nM T33489 CGE4N6 127050301 IC50 = 780 nM T33489 CNEH95 127050311 IC50 = 510 nM T33489 CRHF61 127050469 Ki = 890 nM T33489 CNXM16 127050795 IC50 = 30 nM T33489 C98YZV 127051066 IC50 = 30 nM T33489 C2H6XJ 127051689 IC50 = 30 nM T33489 CO7N6G 127051690 IC50 = 30 nM T33489 CIL98P 127051960 IC50 = 9 nM T33489 C05RTU 127051995 IC50 = 30 nM T33489 C76VSN 127051996 IC50 = 30 nM T33489 CSTM24 127051997 IC50 = 30 nM T33489 CY13OM 127052769 IC50 = 700 nM T33489 CY79KF 127052770 IC50 = 450 nM T33489 C7PX4L 127053168 IC50 = 14 nM T33489 CF6HY4 127053169 IC50 = 400 nM T33489 CH5I8Q 127053170 IC50 = 400 nM T33489 CE97DA 129868496 IC50 = 37800 nM T33489 CC3T4U 135438008 IC50 = 1400 nM T33489 CM5GC3 135712686 IC50 = 4500 nM T33489 C0J4VX 135712687 IC50 = 150 nM T33489 C8ZVB2 135712688 IC50 = 50 nM T33489 CZ62WU 135712689 IC50 = 5000 nM T33489 CMS6C7 135712690 IC50 = 4600 nM T33489 CEH9X6 135712696 IC50 = 250 nM T33489 C05DXY 136100359 IC50 = 16000 nM T33489 CJ73NG 136100360 IC50 = 20000 nM T33489 C9U5ZX 136100361 IC50 = 29000 nM T33489 C2LBA3 136100362 IC50 = 6000 nM T33489 CIY7A3 136100363 IC50 = 8000 nM T33489 CM17NU 136100364 IC50 = 22000 nM T33489 C4BO7N 136100365 IC50 = 18000 nM T33489 CQ6OA3 136100366 IC50 = 3200 nM T33489 CZ8JG0 136100367 IC50 = 25000 nM T33489 C05NHX 136100368 IC50 = 11000 nM T33489 CK57LV 136100369 IC50 = 4000 nM T33489 CV63QC 136100372 IC50 = 50000 nM T33489 C1RH0O 136100377 IC50 = 24000 nM T33489 CXW1R4 136100378 IC50 = 13000 nM T33489 CH3K9T 136100379 IC50 > 100000 nM T33489 C6Z3SV 136100381 IC50 = 15000 nM T33489 C91PTN 136100382 IC50 = 1800 nM T33489 C1XM2Q 136100383 IC50 > 100000 nM T33489 CX09UO 136100384 IC50 = 19000 nM T33489 CC7FR9 136100385 IC50 = 9000 nM T33489 CRP98D 136100386 IC50 > 100000 nM T33489 CXK2Z1 136100387 Ki = 350 nM T33489 C6I7HD 136100388 IC50 = 8000 nM T33489 CIOT59 137631569 IC50 = 360 nM T33489 C25XTW 137632454 IC50 = 123.4 nM T33489 CYD38S 137635650 IC50 = 290 nM T33489 C3G1SO 137636708 IC50 = 3.4 nM T33489 CNB52O 137638205 IC50 = 15.6 nM T33489 CS64RT 137638285 IC50 = 380 nM T33489 CF1PA7 137638452 IC50 = 290 nM T33489 C1FDY3 137640192 IC50 = 244.5 nM T33489 C0Q5AO 137643394 IC50 = 180 nM T33489 CYK0D6 137644698 IC50 = 280 nM T33489 C2XVS3 137645341 IC50 = 440 nM T33489 C5FP6M 137645395 IC50 = 35 nM T33489 CE0OK4 137646056 IC50 = 220.8 nM T33489 CM2PD9 137650549 IC50 = 340 nM T33489 C37GSR 137651543 IC50 = 490 nM T33489 CP0JG8 137654532 IC50 = 260 nM T33489 CPKR15 137656256 IC50 = 2.1 nM T33489 CLZN39 137656380 IC50 = 230 nM T33489 C5YD7K 137658482 IC50 = 300 nM T33489 CB06TQ 137660131 IC50 = 5.1 nM T33489 C37JQW 137660162 IC50 = 210 nM T33489 C67JHC 137660464 IC50 = 180 nM T33489 C62FZT 137661419 IC50 = 105.5 nM T33489 C4CQ7T 155511460 IC50 = 1 nM T33489 C3NJ4C 155511804 IC50 = 14 nM T33489 CITL58 155515974 IC50 = 2.4 nM T33489 CDV32O 155517235 Ki = 350 nM T33489 C2TXG8 155521297 IC50 = 17 nM T33489 C3Z1ER 155524449 IC50 = 0.4 nM T33489 CGLM19 155526670 IC50 = 1 nM T33489 CZ7UV8 155528765 IC50 = 5.1 nM T33489 C3PKZ1 155531378 IC50 = 2.5 nM T33489 CK9OI5 155534879 IC50 = 33.2 nM T33489 CL1S7H 155541009 IC50 = 1 nM T33489 C3VQK7 155542123 IC50 = 0.68 nM T33489 CCA03R 155546507 IC50 = 18.9 nM T33489 C85KFE 155556339 IC50 = 8.8 nM T33489 C7LQI8 155557115 IC50 = 2180 nM T33489 C7MFU2 155558253 IC50 = 43.7 nM T33489 CA29JM 155567815 IC50 = 1690 nM T33489 CDH9L5 155568231 IC50 = 1230 nM T33489 D00AON 9864028 IC50 = 403 nM T33489 D00LFX 20718630 IC50 = 5000 nM T33489 D00OBI 9859866 IC50 = 380 nM T33489 D00OZS 11822292 IC50 = 5900 nM T33489 D01ACT 10858185 IC50 = 13200 nM T33489 D02RJA 44306686 IC50 = 7100 nM T33489 D03NUT 10958461 IC50 = 5000 nM T33489 D03XJE 22733402 IC50 = 260 nM T33489 D04AXP 3001028 IC50 = 7600 nM T33489 D04HNO 44306774 IC50 = 3200 nM T33489 D04YVS 44306753 IC50 = 780 nM T33489 D05KKB 44306687 IC50 = 6900 nM T33489 D05TRN 10018465 IC50 = 500 nM T33489 D06ADL 44306276 IC50 = 5200 nM T33489 D06DVJ 44306759 IC50 = 6900 nM T33489 D06IMK 9729029 IC50 = 4000 nM T33489 D06SMY 10914878 IC50 = 4800 nM T33489 D06YDQ 9796948 IC50 = 3400 nM T33489 D08BTV 135676207 IC50 = 8000 nM T33489 D09BUM 135562887 IC50 = 2300 nM T33489 D09PUF 9842809 IC50 = 30 nM T33489 D09ROV 10367758 Ki = 890 nM T33489 D0AL2D 9885795 IC50 = 190 nM T33489 D0AX3M 9912111 IC50 = 4 nM T33489 D0B1JM 44306292 IC50 = 4800 nM T33489 D0B2XN 9817055 IC50 = 5100 nM T33489 D0D1CV 9879424 IC50 = 3800 nM T33489 D0FH1V 16098588 IC50 = 320 nM T33489 D0G1XC 135529100 IC50 = 460 nM T33489 D0G8HD 44306685 IC50 = 5700 nM T33489 D0I4LL 9861093 IC50 = 16.3 nM T33489 D0L4FM 11030308 IC50 > 10000000 nM T33489 D0M2WG 44306269 IC50 = 4600 nM T33489 D0N8VZ 11583423 IC50 = 1000 nM T33489 D0P6IO 10880277 IC50 = 10500 nM T33489 D0P9ZV 44371205 IC50 = 1700 nM T33489 D0R7QY 127676 IC50 = 0.065 nM T33489 D0S3RZ 9954405 IC50 = 18 nM T33489 D0S5BA 44306775 IC50 = 5000 nM T33489 D0T5OD 10065009 IC50 = 170 nM T33489 D0U7PV 44370998 IC50 = 9300 nM T33489 D0Y9SI 16748617 IC50 = 12000 nM T96235 D00ENY 33032 Ki = 868 nM T96235 D03CNS 2910 EC50 = 3800 nM T96235 D01WBD 9889366 EC50 = 150 nM T96235 D02VKC 3272524 Ki = 600 nM T96235 D03DHQ 148184 EC50 = 156000 nM T96235 D0B0NQ 127894 Ki = 50000 nM T96235 D01PWK 197644 IC50 38000 nM T96235 COC91V 10255 Ki = 1710 nM T96235 C6T4AH 167842 Ki = 457 nM T96235 CC0E1V 447081 Ki = 2.7 nM T96235 CO28NU 447407 EC50 = 7600 nM T96235 CM41VL 656707 EC50 = 520 nM T96235 C1EP3D 2733518 Ki = 11700 nM T96235 CWK7X4 4694356 Ki = 11900 nM T96235 C3JXD9 5289518 EC50 = 20000 nM T96235 C5Z8VG 6324635 Ki > 10000 nM T96235 C9LI7V 9795404 EC50 = 1200 nM T96235 CVW4L3 9795654 Ki = 7.9 nM T96235 COUZ84 9817709 EC50 = 1200 nM T96235 C3OK2F 9840117 EC50 = 5400 nM T96235 CIPQ84 9840720 EC50 = 4000 nM T96235 CFV03Y 9926589 Ki = 262000 nM T96235 CYX24C 9927707 EC50 = 4400 nM T96235 CFC2P8 9928016 EC50 = 290 nM T96235 CJ86VB 10000636 EC50 = 32.8 nM T96235 C97PZI 10000637 EC50 = 22.6 nM T96235 C7Q1MJ 10132082 IC50 > 100000 nM T96235 CRT06M 10199241 EC50 = 551 nM T96235 CRJ2T0 10219992 Ki = 533 nM T96235 C5PD0H 10330442 Ki = 5600 nM T96235 CFKJ76 10352480 Ki = 182 nM T96235 C7GIJ3 10398361 Ki = 4710 nM T96235 C1N2VM 10420002 Ki = 1055 nM T96235 C7B9RP 10494940 EC50 = 19600 nM T96235 C67UMV 10519128 EC50 = 2000 nM T96235 C2O5ZN 10520589 EC50 = 130 nM T96235 CXE7F5 10541731 Ki > 10000 nM T96235 CH35TY 10547998 EC50 > 100000 nM T96235 C12XCT 10567789 EC50 = 7200 nM T96235 CNT0K7 10571414 EC50 > 100000 nM T96235 CO87ST 10617783 EC50 > 100000 nM T96235 C8F5UO 10618573 EC50 = 32900 nM T96235 CI5R2A 10620266 EC50 > 100000 nM T96235 C2UO7I 10643804 EC50 > 3000 nM T96235 C0O6ZI 10658567 EC50 = 3000000 nM T96235 C3GOV7 10660661 EC50 = 12800 nM T96235 C0TH7D 10680928 EC50 > 100000 nM T96235 CZ0U2V 10685310 EC50 = 4500 nM T96235 CT9KQ0 10713611 EC50 = 1400 nM T96235 CH4L8X 10737832 EC50 = 62500 nM T96235 C4EHX7 10783025 EC50 = 23800 nM T96235 CJG4F8 10783725 EC50 = 250 nM T96235 CJ76SM 10784150 EC50 > 3000 nM T96235 CRDQ31 10829310 EC50 = 1000 nM T96235 CQ3GE5 10829935 EC50 = 27900 nM T96235 CN85QA 10853988 EC50 = 270 nM T96235 CY4MV7 10935011 EC50 = 621 nM T96235 CJ3QY6 10967953 EC50 = 434 nM T96235 CHW4K6 10968688 EC50 = 1100 nM T96235 CG0T8R 11033972 EC50 = 247 nM T96235 CJZ04V 11096831 Ki = 207 nM T96235 CNTE47 11119059 EC50 = 1740 nM T96235 C1KNU5 11120538 EC50 = 190 nM T96235 CW0LO5 11121532 EC50 = 68 nM T96235 CQ97KS 11198294 EC50 = 213 nM T96235 CQ38WM 11219775 Ki = 732 nM T96235 CGRT02 11288627 Ki = 44.4 nM T96235 C2EA6X 11291212 EC50 = 53 nM T96235 CY43TM 11748700 EC50 = 118 nM T96235 CM1GA4 11773296 EC50 = 77 nM T96235 C4Q5VR 11782933 EC50 = 82.1 nM T96235 CHUX80 11818375 Ki = 2350 nM T96235 CDGZ79 11820131 Ki = 10300 nM T96235 CG3M6R 11833226 EC50 = 403 nM T96235 C3F4KH 16046205 EC50 = 214 nM T96235 CX2VU6 16046206 EC50 = 183 nM T96235 CQ2YP8 16659202 EC50 = 75000 nM T96235 C4U7OS 44152410 Ki = 451 nM T96235 CFZS21 44307184 EC50 = 520 nM T96235 CW9TR7 44346780 Ki = 3.6 nM T96235 C64ELF 44346789 Ki = 89 nM T96235 CQJW06 44346790 Ki = 189 nM T96235 C15MPO 44346798 Ki = 19.9 nM T96235 CE8F0R 44416383 EC50 = 440 nM T96235 CS73PO 44416384 EC50 = 2892 nM T96235 CS0G6A 44416385 EC50 = 1873 nM T96235 CVW13Z 44416400 EC50 > 3000 nM T96235 C70TDS 44416401 EC50 = 489 nM T96235 C73EAN 44416520 EC50 = 795 nM T96235 COQ86N 44416680 EC50 = 629 nM T96235 C84BWG 44416681 EC50 = 474 nM T96235 CBW5D3 44416682 EC50 = 1009 nM T96235 CAYR16 44416702 EC50 = 273 nM T96235 CXN16F 44416703 EC50 > 3000 nM T96235 C60GWQ 44416732 EC50 = 554 nM T96235 C1YW8F 44416748 EC50 = 394 nM T96235 C4NDM6 44416749 EC50 = 1979 nM T96235 CHD28J 44416750 EC50 > 3000 nM T96235 CQD2Y3 44416776 EC50 = 1143 nM T96235 CIQ92O 44416794 EC50 = 2085 nM T96235 C2YR8D 44416795 EC50 = 790 nM T96235 CIRK69 44416811 EC50 = 738 nM T96235 CCZW78 44416812 EC50 = 1051 nM T96235 CE2NL6 44416834 EC50 = 386 nM T96235 CVC38F 44416870 EC50 = 619 nM T96235 C7PW9S 44416873 EC50 = 373 nM T96235 CAGW51 44416888 EC50 > 3000 nM T96235 C3ZIJ2 44416889 EC50 > 3000 nM T96235 CGH79E 44416892 EC50 = 631 nM T96235 CIW5X0 44416905 EC50 = 679 nM T96235 CRB28F 44416986 EC50 = 146 nM T96235 CD3G7X 44417019 EC50 = 242 nM T96235 CD7JY5 44417039 EC50 = 223 nM T96235 CJS5Z7 44417040 EC50 = 80 nM T96235 CP71ZU 44417062 EC50 = 910 nM T96235 CPNL12 44417063 EC50 = 1082 nM T96235 CYQ4C9 44417081 EC50 = 532 nM T96235 CK8FI3 44417082 EC50 = 157 nM T96235 C56NLW 127039193 EC50 = 100000 nM T96235 C1G7SF 127039194 EC50 = 55000 nM T96235 C5Q6ZI 137638800 Ki = 7400 nM T96235 C03KAU 155519563 EC50 > 1000000 nM T96235 CM4AJ5 155545606 EC50 = 34673.69 nM T96235 CBS42U 155557317 EC50 = 51000 nM T96235 D01DMS 447196 Ki = 972 nM T96235 D03RGP 1221 Ki = 40 nM T96235 D04SMQ 440053 Ki = 8850 nM T96235 D09LXQ 126569 Ki = 305 nM T96235 D0C5WK 9873570 EC50 = 660 nM T96235 D0KD6O 5288598 EC50 = 15000 nM T96235 D0N1CL 9799478 IC50 > 100000 nM T96235 D0O7OE 122294 IC50 = 430 nM T96235 D0T5SU 158397 Ki = 40 nM T53469 D0J3SU 9847835 Ki > 5000 nM T53469 CV7IN2 104934 Ki = 337 nM T53469 C1KR5B 5327301 Ki = 96000 nM T53469 C37TKL 5327302 Ki = 21000 nM T53469 C64ZMN 5327304 Ki = 92000 nM T53469 C3IZ2W 5327307 Ki = 13000 nM T53469 C16DTL 5327308 Ki = 38000 nM T53469 C4O3QY 5327309 Ki > 100000 nM T53469 C3GUM7 5327310 Ki = 27000 nM T53469 CFN2P6 9800285 Ki = 30000 nM T53469 C4XO3K 9821545 Ki = 33000 nM T53469 CLAC59 9828058 Ki = 248 nM T53469 C6S3KT 9840223 Ki > 25000 nM T53469 CX67SZ 10826725 Ki = 5000 nM T53469 CDX7A4 10963183 Ki = 22000 nM T53469 CDT9G3 11467504 IC50 = 0.5 nM T53469 CJ57OA 14585243 Ki = 207 nM T53469 C25ELB 44143088 IC50 = 33113.11 nM T53469 CD8WB9 44304162 Ki > 50000 nM T53469 C8D5TB 44364680 Ki = 38000 nM T53469 C86ORE 44459987 IC50 = 8128.31 nM T53469 CDY2W5 49796910 IC50 = 0.3 nM T53469 CGY3W2 71471109 IC50 = 510 nM T53469 CANH70 71716242 IC50 = 5600 nM T53469 C40WIR 71718085 IC50 = 180 nM T53469 CU75VK 71719897 IC50 = 370 nM T53469 CBV6F1 71720507 IC50 = 90 nM T53469 CID3N6 134134572 IC50 > 5000 nM T53469 CV0R3B 134135432 Ki = 267 nM T53469 C3D7LQ 134136688 Ki = 870 nM T53469 CBY95D 134138690 IC50 > 5000 nM T53469 CG3EI1 134145896 Ki = 148 nM T53469 CI9X3K 134147411 Ki = 8 nM T53469 CP16IA 134148745 Ki = 276 nM T53469 CPE90G 134149983 Ki = 393 nM T53469 CBE39C 134151245 Ki = 563 nM T53469 CY0LD4 134152014 Ki = 306 nM T53469 C3K5HR 134153309 Ki = 119 nM T53469 CWQT79 134156687 Ki = 215 nM T53469 D0N5MU 4117381 Ki > 50000 nM T53469 D0Q9XX 515950 Ki = 4000 nM T53469 D0Y5IQ 44255320 IC50 = 5000 nM T05114 D0SH3I 387447 IC50 = 1190 nM T05114 D0V3YT 10324367 IC50 = 32 nM T05114 D0X9CH 3010818 IC50 = 26 nM T05114 D00LOB 9866964 Ki > 26000 nM T05114 D01YIO 10146470 Ki = 2.3 nM T05114 D0VO0T 24800541 IC50 = 3530 nM T05114 C3MV6U 87111 IC50 = 340000 nM T05114 CP9FG4 99625 IC50 = 400 nM T05114 CH67RW 152801 IC50 > 1000000 nM T05114 CFG3E0 321710 IC50 > 1000000 nM T05114 CN0XJ3 439647 IC50 = 3300 nM T05114 CY84OK 603829 IC50 = 90000 nM T05114 C05EGK 736344 IC50 = 470000 nM T05114 C18MHT 1480686 IC50 > 1000000 nM T05114 CK32XJ 2773289 IC50 = 570000 nM T05114 CDNF82 2824428 IC50 = 10600 nM T05114 C94TLN 3731010 IC50 > 1000000 nM T05114 CW9DQ2 4476325 Ki = 2.3 nM T05114 C7Q4ZX 6106643 IC50 = 12000 nM T05114 CANW64 9798519 IC50 = 380 nM T05114 CMUY79 9800909 IC50 = 22 nM T05114 C92QSE 9801235 IC50 > 100000 nM T05114 CD8G1T 9818360 IC50 = 6200 nM T05114 C9NHA3 9821476 IC50 = 300 nM T05114 C7UKF5 9825353 IC50 = 56 nM T05114 CGNB60 9830581 IC50 = 27 nM T05114 C5T0GJ 9895523 IC50 = 20 nM T05114 CGL12S 9916581 Ki = 2.62 nM T05114 CIQX83 9938207 Ki = 1.12 nM T05114 C0WT4P 10024711 IC50 = 20 nM T05114 CHT4F7 10032234 Ki = 3 nM T05114 C03GYH 10058155 IC50 > 1000000 nM T05114 CE7LT8 10086155 IC50 = 30000 nM T05114 CD6KX7 10162462 IC50 = 203 nM T05114 CSR74M 10228660 IC50 > 100000 nM T05114 CB09RG 10258388 IC50 = 6 nM T05114 CFX95N 10259109 Ki = 1.3 nM T05114 CE8YI4 10316093 IC50 = 0.85 nM T05114 CRP54X 10364794 IC50 = 23 nM T05114 C9M3VF 10366027 IC50 = 82 nM T05114 CCQA34 10383086 IC50 = 360 nM T05114 CEPM12 10391460 IC50 = 220 nM T05114 CCL85B 10394816 IC50 = 270 nM T05114 C2UNX1 10407325 IC50 = 35 nM T05114 CVB41T 10416916 Ki = 5.6 nM T05114 CORP79 10431323 IC50 = 22 nM T05114 CBIN45 10444299 IC50 = 1700 nM T05114 C3EN8D 10479280 Ki = 50.6 nM T05114 C9M7CE 10497407 IC50 = 40 nM T05114 CYC5G6 10497621 IC50 = 30 nM T05114 CJN97A 10499538 IC50 = 60 nM T05114 CC1PL9 10504801 Ki = 3850 nM T05114 C6D3UM 10504812 IC50 = 510000 nM T05114 C4N9CG 10505462 Ki = 90.7 nM T05114 CI56MJ 10505892 Ki = 125 nM T05114 C4XU1H 10505893 Ki = 489 nM T05114 CG1N3Z 10506615 Ki = 12 nM T05114 CAMR48 10506883 Ki = 5.57 nM T05114 C6M3GF 10506968 Ki = 76 nM T05114 COKF15 10520443 IC50 = 2600 nM T05114 CIMX79 10524714 IC50 = 170 nM T05114 C5LR1J 10527210 IC50 = 28000 nM T05114 C0DV7Q 10528861 Ki > 10000 nM T05114 C3VQM6 10529952 IC50 = 3200 nM T05114 CX6WB8 10531400 Ki = 26.1 nM T05114 C5F6RU 10531565 Ki = 9.32 nM T05114 CF7A0S 10531953 Ki = 3.56 nM T05114 CTN78E 10545533 IC50 = 550 nM T05114 CCE5M4 10551184 IC50 = 900 nM T05114 C3UPR0 10554476 Ki = 16.9 nM T05114 CZ53TL 10554981 Ki = 5.6 nM T05114 CZL85V 10572734 IC50 = 100000 nM T05114 CHAT84 10577682 Ki = 60.6 nM T05114 C2BRT9 10578876 Ki = 44.2 nM T05114 CNL0X1 10578948 Ki = 56.3 nM T05114 C20JKT 10593313 IC50 = 68 nM T05114 CZ8PK9 10599803 IC50 = 170 nM T05114 C2V4IZ 10616405 IC50 > 100000 nM T05114 C9I3QE 10616695 IC50 = 370 nM T05114 CS52KZ 10617888 IC50 = 1100 nM T05114 C38SDV 10619385 IC50 = 29 nM T05114 C83JQD 10620089 IC50 = 18 nM T05114 C4K1BD 10620298 IC50 = 5000 nM T05114 C5X0QT 10625780 IC50 = 150 nM T05114 CZ23TH 10627192 Ki = 174 nM T05114 CUX7N1 10627346 Ki = 41.8 nM T05114 CH06SV 10627450 Ki = 16.6 nM T05114 C0TQJ4 10627517 Ki = 10.2 nM T05114 C8BVH0 10627562 Ki = 59.5 nM T05114 C6V4NJ 10642042 IC50 = 35000 nM T05114 CA9XC0 10647781 Ki = 589 nM T05114 CS0WB7 10649867 Ki = 93.1 nM T05114 CPNI68 10650491 Ki = 32.5 nM T05114 CM57UY 10666214 IC50 = 5900 nM T05114 CBL23T 10674706 Ki = 15.7 nM T05114 C4FP2G 10674707 Ki = 440 nM T05114 C8QB4K 10689926 IC50 = 700 nM T05114 CVS68A 10697425 Ki = 183 nM T05114 CZ57RO 10697572 IC50 = 62000 nM T05114 C2WC3O 10698015 Ki = 23 nM T05114 C1WV6C 10698103 Ki = 84.7 nM T05114 C63JIQ 10698344 Ki = 16.9 nM T05114 C5V6IF 10698497 Ki = 68.6 nM T05114 CF1HZ7 10698873 Ki = 9.7 nM T05114 C6S2JY 10712874 IC50 = 130 nM T05114 CFCP28 10714430 IC50 = 82 nM T05114 CP7Y9Z 10714544 IC50 = 110 nM T05114 CPT0M6 10715096 IC50 = 66 nM T05114 CE7CB3 10715299 IC50 = 500 nM T05114 C04SDQ 10720538 Ki > 10000 nM T05114 CT42IS 10721198 Ki = 73.3 nM T05114 CD0I2U 10736348 IC50 = 580 nM T05114 CX9JY3 10737216 IC50 = 860 nM T05114 C06EQF 10739429 IC50 = 65000 nM T05114 CVX58I 10740202 IC50 = 700 nM T05114 C8OKL4 10745283 Ki = 43.5 nM T05114 CP51CW 10745318 Ki = 94 nM T05114 C1TB8N 10764081 IC50 = 14000 nM T05114 C3MH6G 10765640 IC50 = 3300 nM T05114 CW92LC 10768479 Ki = 182 nM T05114 CMF61Y 10770047 Ki = 33.7 nM T05114 C4J2AM 10782637 IC50 = 1800 nM T05114 CFR3G8 10792830 Ki = 18.5 nM T05114 CKV52E 10792972 Ki = 74.3 nM T05114 CUFX71 10793116 Ki = 7.71 nM T05114 CEIV70 10793518 Ki = 13.8 nM T05114 CSO9H0 10811389 IC50 > 100000 nM T05114 C4T9US 10816519 Ki = 77.4 nM T05114 CL85VD 10835279 IC50 = 800 nM T05114 CX3E7A 10838826 IC50 = 19000 nM T05114 CR82DN 10839877 Ki = 2120 nM T05114 CYBQ47 10841038 Ki = 30 nM T05114 C27IBH 11154988 IC50 = 11 nM T05114 CZ7V9G 11223476 IC50 = 50 nM T05114 C39NQW 11235804 IC50 = 29 nM T05114 CG59UY 11236464 Ki = 11 nM T05114 CZ1OD3 11270172 IC50 = 16 nM T05114 CS4Y2X 11303525 IC50 = 920 nM T05114 C9QSZ3 11305284 IC50 = 58 nM T05114 CF6P9Z 11316579 IC50 = 21 nM T05114 CY3RT6 11318361 IC50 = 240 nM T05114 C9R7BV 11350018 IC50 = 120 nM T05114 CF25UN 11350795 IC50 = 66 nM T05114 C56LCG 11373688 IC50 = 10 nM T05114 CO4PX8 11385226 IC50 = 160 nM T05114 CV1ID6 11429319 IC50 = 90 nM T05114 C92OWP 11453143 IC50 = 13 nM T05114 CPW41T 11453471 IC50 = 3.5 nM T05114 C1H6AR 11486613 IC50 = 60 nM T05114 CF5Q4A 11487223 IC50 = 80 nM T05114 CLAK97 11540629 IC50 = 300 nM T05114 C93USP 11626693 IC50 = 34 nM T05114 C07MTY 11634767 IC50 = 170 nM T05114 C1ZK9V 11684537 IC50 = 240 nM T05114 C6RY7J 11725023 IC50 = 300 nM T05114 CKOV89 11799023 Ki = 13.3 nM T05114 C1CQS5 11800896 Ki = 10.2 nM T05114 C0GZD9 11801158 Ki = 14.3 nM T05114 CC53TD 12043588 IC50 = 710 nM T05114 C15CLN 12045136 IC50 = 880 nM T05114 CTJ72A 12045140 IC50 = 305 nM T05114 CE5O3V 12222540 IC50 = 2 nM T05114 C93MAZ 12222541 IC50 = 2.3 nM T05114 CYGX75 12496475 IC50 > 1000000 nM T05114 C7C1GX 12972072 IC50 = 550 nM T05114 C2QCF6 12972074 IC50 = 19 nM T05114 C9C5WP 12972379 IC50 = 140 nM T05114 CY9X8B 12972381 IC50 = 1600 nM T05114 CH4B2E 12972382 IC50 = 50 nM T05114 CH7SX5 12972383 IC50 = 70 nM T05114 CDNM15 13224504 IC50 = 300 nM T05114 C0QXL9 13224509 IC50 = 1400 nM T05114 C10ALY 13339657 IC50 = 1300 nM T05114 C2DGN3 14046022 IC50 = 40000 nM T05114 C19ARJ 15984063 Ki > 150000 nM T05114 CRV3H2 16204287 IC50 = 190 nM T05114 C4B2DO 16204288 IC50 = 2500 nM T05114 C46PRL 16204387 IC50 = 210 nM T05114 C0P6CM 16204388 IC50 = 2100 nM T05114 C43SRY 16204391 IC50 = 280 nM T05114 CE1P9X 16204392 IC50 = 165 nM T05114 C2ORE0 16204393 IC50 = 10400 nM T05114 C74DEI 17855420 IC50 > 1000 nM T05114 COE8A7 17878496 IC50 = 18 nM T05114 CELQ36 21953543 IC50 > 1000000 nM T05114 CKR24L 22041443 IC50 = 337 nM T05114 CB53MJ 22041451 IC50 = 159 nM T05114 CI08KO 22041455 IC50 = 325 nM T05114 C6DGB9 22041474 IC50 = 663 nM T05114 C1Z9SX 24776379 IC50 > 5000 nM T05114 CCG0Z2 25124204 IC50 = 25 nM T05114 CL0M7R 44143089 IC50 = 89125.09 nM T05114 C3XVB5 44291692 IC50 = 40000 nM T05114 C36TCK 44291947 IC50 = 48 nM T05114 C65TOU 44303193 IC50 = 15000 nM T05114 C2DM3E 44303204 IC50 = 4700 nM T05114 C9N4KA 44303215 IC50 = 2100 nM T05114 CE3NJ0 44303216 IC50 = 730 nM T05114 C3E6HC 44303217 IC50 = 2200 nM T05114 CR68VO 44303218 IC50 = 3100 nM T05114 CR6GO9 44303240 IC50 = 2700 nM T05114 C6YB7J 44303242 IC50 = 600 nM T05114 CWOM61 44303259 IC50 = 3700 nM T05114 C0C8FX 44303260 IC50 = 890 nM T05114 CWUI78 44303375 IC50 = 780 nM T05114 CJ15HX 44303391 IC50 = 1800 nM T05114 CH6TE7 44303392 IC50 = 1900 nM T05114 CVJS18 44303415 IC50 = 430 nM T05114 C1W6MX 44303477 IC50 = 2500 nM T05114 CSB6M5 44303496 IC50 = 1200 nM T05114 CGNR45 44303533 IC50 = 1200 nM T05114 CTRX10 44303534 IC50 = 2400 nM T05114 C20OYT 44303535 IC50 = 890 nM T05114 C1Y2QB 44303536 IC50 = 2200 nM T05114 CGP52Y 44303588 IC50 = 1400 nM T05114 CH13CK 44303589 IC50 = 2500 nM T05114 CQ82JC 44303644 IC50 = 1900 nM T05114 CO3V6E 44303657 IC50 = 400 nM T05114 C5L1DC 44308976 IC50 = 27000 nM T05114 CM2N3I 44316444 IC50 = 70 nM T05114 CICF46 44316445 IC50 = 430 nM T05114 CYJ9N2 44316484 IC50 = 170 nM T05114 CKN8C1 44316486 IC50 = 6 nM T05114 CDZ2K1 44316507 IC50 = 4000 nM T05114 CX08UQ 44316508 IC50 = 440 nM T05114 CUE40X 44316655 IC50 = 50 nM T05114 C2WF1Q 44316715 IC50 = 1650 nM T05114 C6RW9G 44316735 IC50 > 10000 nM T05114 CSAF06 44316754 IC50 = 150 nM T05114 CW90JQ 44316764 IC50 = 250 nM T05114 C61COX 44316919 IC50 > 10000 nM T05114 C8Z3GE 44317096 IC50 = 410 nM T05114 COUN74 44317097 IC50 = 6800 nM T05114 CT3OS4 44317111 IC50 > 10000 nM T05114 CE03NG 44317159 IC50 > 10000 nM T05114 C2GV6C 44317160 IC50 = 300 nM T05114 C5SQ3Y 44317185 IC50 = 3500 nM T05114 CDO29P 44317186 IC50 = 1700 nM T05114 CD7K3O 44317187 IC50 = 7310 nM T05114 CM7N0R 44317231 IC50 = 24 nM T05114 CT9C5P 44317320 IC50 = 15600 nM T05114 CJI97E 44317349 IC50 = 11000 nM T05114 CTEC69 44317399 IC50 = 37 nM T05114 C2LEB8 44317400 IC50 = 57 nM T05114 C1L0GY 44317409 IC50 = 26 nM T05114 CIP4C9 44353215 IC50 = 154 nM T05114 C10JVQ 44353225 IC50 > 1000 nM T05114 C30TRA 44353235 IC50 > 1000 nM T05114 C9LP4D 44353342 IC50 = 1647 nM T05114 C0LZH1 44353420 IC50 = 192 nM T05114 C0RI4F 44353490 IC50 = 594 nM T05114 CV9P4O 44353491 IC50 = 4208 nM T05114 CDLQ89 44354931 IC50 = 58 nM T05114 CZG9E2 44354934 IC50 = 3000 nM T05114 C7NWU8 44354935 IC50 = 29000 nM T05114 C5UJB8 44354936 IC50 = 5 nM T05114 CRL78E 44354968 IC50 = 5.6 nM T05114 CM73HF 44354971 IC50 = 37 nM T05114 CVYF38 44354984 IC50 = 47000 nM T05114 CZDW93 44355000 IC50 = 13000 nM T05114 CG1VN6 44355001 IC50 = 8700 nM T05114 CL04TR 44355071 IC50 = 130 nM T05114 C9U4BR 44355072 IC50 = 13 nM T05114 CI4R1U 44355083 IC50 = 32 nM T05114 CDON50 44355100 IC50 > 1000000 nM T05114 C34UGZ 44366594 Ki = 55.8 nM T05114 C6ENF2 44382957 Ki = 14.2 nM T05114 CS6UN7 44383119 Ki = 13.1 nM T05114 C3S8JB 44383120 Ki = 1550 nM T05114 C7H1KL 44383138 Ki = 6.3 nM T05114 CM3L2E 44383139 Ki = 6.8 nM T05114 CW4Y2G 44383169 Ki = 6.5 nM T05114 CCFH08 44383170 Ki = 7.1 nM T05114 CZ45AF 44383171 Ki = 3.1 nM T05114 CF19SJ 44383172 Ki = 16.5 nM T05114 C32VXU 44383175 Ki = 513 nM T05114 CP0YT7 44383405 Ki = 5.6 nM T05114 CBP42U 44383406 Ki = 3.9 nM T05114 C4A5HG 44383407 Ki = 27.5 nM T05114 CAT06Q 44383408 Ki = 70.1 nM T05114 C24RJS 44383410 Ki = 30.1 nM T05114 CKQR02 44383458 Ki = 7.4 nM T05114 CZ73PA 44383459 Ki = 28.7 nM T05114 CRGZ24 44383473 Ki = 6.7 nM T05114 C03GUY 44383483 Ki = 6 nM T05114 CV6M2L 44383625 Ki = 493 nM T05114 CR82ID 44383626 Ki = 65.6 nM T05114 C54FTU 44383779 Ki = 18.3 nM T05114 C56OZS 44383818 Ki = 16.3 nM T05114 CCJT53 44383923 Ki = 24 nM T05114 C8I7UK 44383924 Ki = 36.4 nM T05114 CBW62J 44383984 Ki = 12.5 nM T05114 C2Y4OV 44384261 Ki = 3620 nM T05114 CIK29L 44384262 Ki = 1040 nM T05114 CD7C8F 44384263 Ki = 1010 nM T05114 C9K5XD 44384375 Ki = 21.1 nM T05114 CD98YX 44384376 Ki = 36.6 nM T05114 CC2LZ6 44384377 Ki = 22.8 nM T05114 C3BX5Y 44412781 Ki > 150000 nM T05114 C50KCG 44439950 IC50 = 420 nM T05114 C7HQ3R 44439951 IC50 = 1500 nM T05114 C2JIB9 44439952 IC50 > 10000 nM T05114 CM1AF3 44439953 IC50 > 10000 nM T05114 C5IVE4 44439954 IC50 > 10000 nM T05114 CTV73R 44439955 IC50 > 10000 nM T05114 C87GWX 44439956 IC50 = 460 nM T05114 C8IGC1 44439957 IC50 = 310 nM T05114 CP1Z9O 44439958 IC50 = 110 nM T05114 CRJ2V3 44439959 IC50 = 150 nM T05114 CY6G1J 44439961 IC50 = 140 nM T05114 C3CT0V 44439962 IC50 = 180 nM T05114 C8M6UP 44439963 IC50 = 83 nM T05114 C7AXP5 44439964 IC50 = 220 nM T05114 C8K2PE 44439965 IC50 = 280 nM T05114 CN16CB 44439967 IC50 = 42 nM T05114 CGT8B4 44439968 IC50 = 26 nM T05114 CM8Q6V 44439969 IC50 = 27 nM T05114 CC5V2F 44439970 IC50 = 1100 nM T05114 C5YLN8 44439971 IC50 = 7400 nM T05114 C5EW2F 44439972 IC50 = 23 nM T05114 CA7V6O 44439973 IC50 = 4200 nM T05114 CK0M2A 44439974 IC50 = 27 nM T05114 CMHZ07 44439975 IC50 > 10000 nM T05114 CZ78KW 44440009 IC50 = 34 nM T05114 CQ64GY 44440010 IC50 = 4900 nM T05114 CSGK96 44440011 IC50 > 100000 nM T05114 CMI5D7 44440014 IC50 = 44500 nM T05114 CYZ6V9 44440019 IC50 = 5300 nM T05114 C84HKM 44440020 IC50 = 2800 nM T05114 CBV73O 44440021 IC50 = 3000 nM T05114 C93UJB 44440022 IC50 = 69300 nM T05114 CDX4W5 44440023 IC50 > 100000 nM T05114 CJLN69 44440024 IC50 = 470 nM T05114 C9WQ2P 44440025 IC50 = 2500 nM T05114 CP17KC 44440026 IC50 = 460 nM T05114 C3GTR1 44440027 IC50 = 340 nM T05114 CJ9CQ7 44440030 IC50 = 540 nM T05114 CQF34M 44440032 IC50 = 2600 nM T05114 C30EBQ 44440034 IC50 = 410 nM T05114 C02DTK 44440035 IC50 = 630 nM T05114 CH2B9R 44440066 IC50 > 10000 nM T05114 CK73VI 44440078 IC50 > 10000 nM T05114 CG05SO 44440082 IC50 > 10000 nM T05114 C0M4NO 44453158 Ki = 23 nM T05114 CP1WH2 44453159 Ki = 5.6 nM T05114 C0RLW3 44453160 Ki = 4.8 nM T05114 CO3J1P 44453194 Ki = 73 nM T05114 C24UMT 44453196 Ki = 590 nM T05114 CV26YQ 44453221 Ki = 120 nM T05114 C19PXD 44453223 Ki = 3800 nM T05114 CNG12O 44453224 Ki = 180 nM T05114 CVI8H9 44459742 Ki = 28.9 nM T05114 C2PVE0 45103523 Ki > 26000 nM T05114 CGN14R 45103723 Ki > 26000 nM T05114 C4YAJ7 46228924 IC50 > 10000 nM T05114 CO6F3U 53249965 IC50 = 97 nM T05114 C84YEG 53322017 IC50 = 3.1 nM T05114 C08CBG 53326855 IC50 = 0.46 nM T05114 C87EBD 54684614 IC50 = 0.42 ug.mL-1 T05114 CS48GW 54687215 IC50 = 0.25 ug.mL-1 T05114 C8U4OD 56649692 IC50 > 1000000 nM T05114 CY3IO1 56659828 IC50 = 4200 nM T05114 CI2AB4 56663296 IC50 = 620 nM T05114 CT2G3R 56666720 IC50 = 70 nM T05114 CQH46K 56666721 IC50 = 600 nM T05114 C3V0AU 56666722 IC50 = 2800 nM T05114 CZ3O2H 56670144 IC50 = 570 nM T05114 CNL70Y 56670149 IC50 = 65 nM T05114 C0HJL7 56673658 IC50 = 170 nM T05114 CP5B7A 56673659 IC50 = 640 nM T05114 CE58OY 56673664 IC50 = 140 nM T05114 C9F5UR 56676983 IC50 > 10000 nM T05114 CL9XA8 56680306 IC50 > 10000 nM T05114 CHNX69 56680307 IC50 = 640 nM T05114 CP3IV1 56680314 IC50 = 220 nM T05114 CSF9P8 56683631 IC50 = 1900 nM T05114 CD57KP 56683632 IC50 = 2600 nM T05114 CP1MR2 56683633 IC50 > 10000 nM T05114 CG7O3N 56683634 IC50 = 280 nM T05114 C8UHN3 56949979 IC50 > 100000 nM T05114 CAX5L0 57670920 IC50 = 4200 nM T05114 CU1EV2 57670929 IC50 = 3700 nM T05114 C7W9RJ 57670947 IC50 = 1200 nM T05114 CY21OJ 57670988 IC50 = 570 nM T05114 C78OCT 57670989 IC50 = 1600 nM T05114 C3RW2I 57670992 IC50 = 3000 nM T05114 CJSM52 57670996 IC50 = 2000 nM T05114 C63WDM 57670998 IC50 = 1000 nM T05114 C10KLT 57671006 IC50 = 380 nM T05114 C7U0IW 57671011 IC50 = 5200 nM T05114 CJV9Y2 57671028 IC50 = 790 nM T05114 CR3PD4 57671034 IC50 = 3100 nM T05114 C0UIF5 57671050 IC50 = 380 nM T05114 CC6GT9 57671056 IC50 = 730 nM T05114 CPLB43 57671061 IC50 = 570 nM T05114 CQ7C0H 57671074 IC50 = 8500 nM T05114 C67FPY 57671083 IC50 = 2770 nM T05114 CZ8B1P 57671099 IC50 = 2600 nM T05114 CX9NI4 57671100 IC50 = 520 nM T05114 CY26NE 57671116 IC50 = 660 nM T05114 CA6HT0 57671121 IC50 = 1300 nM T05114 C9E6CB 57671131 IC50 = 260 nM T05114 CE50SP 57671142 IC50 = 2800 nM T05114 CMY4H9 57671144 IC50 = 850 nM T05114 CJO75X 57671161 IC50 = 570 nM T05114 CO29GJ 57671167 IC50 = 770 nM T05114 CF2Q3E 59497392 IC50 = 240 nM T05114 C2W3AK 59497404 IC50 = 2300 nM T05114 C0E1KN 59497528 IC50 = 40 nM T05114 CAWN80 59497611 IC50 = 3800 nM T05114 CSQY41 59497643 IC50 = 50 nM T05114 C31NTK 59497690 IC50 = 60 nM T05114 C50MEH 71682307 IC50 = 1400 nM T05114 CO8PQ5 71682308 IC50 = 1500 nM T05114 C78DJQ 71711730 IC50 < 10000 nM T05114 CL23VT 71723878 IC50 = 410 nM T05114 CR4MN6 71724022 IC50 = 1640 nM T05114 C1CDP8 73351764 Ki = 82.1 nM T05114 CDX49U 73355024 IC50 = 3900 nM T05114 C6TO7X 86672192 IC50 = 8.9 nM T05114 CS4M5B 88994359 IC50 = 2400 nM T05114 C0FC3W 88994460 IC50 = 78 nM T05114 C1F4RI 88994537 IC50 = 240 nM T05114 CLB96T 88994717 IC50 = 1200 nM T05114 C6JI5X 88994760 IC50 = 580 nM T05114 C54RKQ 88994878 IC50 = 50 nM T05114 C8WS7U 137646736 Ki = 590 nM T05114 C2D6KY 137650380 Ki = 490 nM T05114 CE3D8P 145951877 IC50 = 101000 nM T05114 CL42TO 145953024 IC50 = 23200 nM T05114 CK80JP 155515537 Ki = 37 nM T05114 CS91KQ 155515771 Ki = 10 nM T05114 C0BDN1 155520910 Ki = 64 nM T05114 CW1B5Z 155521967 Ki = 1.7 nM T05114 CBU5W0 155524880 IC50 > 10000 nM T05114 C4QT3M 155526246 Ki = 6.6 nM T05114 CVX87F 155529349 Ki = 740 nM T05114 CAX56B 155530871 Ki = 54 nM T05114 C2X5EJ 155531124 Ki = 2.2 nM T05114 CPC60R 155533917 Ki = 20 nM T05114 C8Z2YM 155534914 IC50 > 5000 nM T05114 CSX02D 155535809 IC50 > 10000 nM T05114 CFAW67 155552500 IC50 > 5000 nM T05114 C2E5GR 155554478 IC50 > 10000 nM T05114 CE3G5W 155556110 Ki = 19 nM T05114 C0SND3 155557259 Ki = 54 nM T05114 CTS63Q 155558248 Ki = 1.8 nM T05114 CFX07G 155558369 IC50 > 10000 nM T05114 C2K6ER 155558569 Ki = 11 nM T05114 C5R4VY 155566937 Ki = 5.7 nM T05114 CO8GJ3 155568502 Ki = 7.5 nM T05114 CT8EM4 155568853 Ki = 1700 nM T05114 CU62EW 155568945 Ki = 0.22 nM T05114 D05ICF 3492365 IC50 = 140 nM T05114 D08QZD 9829503 Ki = 3.68 nM T05114 D0C8UF 44439966 IC50 = 39 nM T05114 D0F2YC 10038543 IC50 = 4 nM T05114 D0L0QR 443119 IC50 = 9.36 nM T05114 D0Y5IQ 44255320 IC50 = 10000 nM T68876 D00ENY 33032 Ki = 789 nM T68876 D02VKC 3272524 Ki = 18000 nM T68876 D0B0NQ 127894 Ki > 100000 nM T68876 COC91V 10255 Ki = 10 nM T68876 C5Z8VG 6324635 Ki = 617 nM T68876 C2L6EK 9807075 Ki = 1400 nM T68876 C9TLQ4 9861035 Ki = 423 nM T68876 CG0WB9 9958244 Ki = 680 nM T68876 CRJ2T0 10219992 Ki = 5730 nM T68876 C5PD0H 10330442 Ki = 518 nM T68876 C7GIJ3 10398361 Ki = 12400 nM T68876 CX1V3L 10437436 Ki = 46 nM T68876 CXE7F5 10541731 Ki = 42 nM T68876 C8V4UC 11544633 Ki = 111000 nM T68876 CHO09Z 11674376 Ki = 374000 nM T68876 CDGZ79 11820131 Ki = 10500 nM T68876 C0YK6J 22100077 Ki = 5700 nM T68876 CM9D7U 22100122 Ki = 530 nM T68876 CIG65E 22449297 Ki = 4100 nM T68876 CJ5X0B 44307207 Ki = 1400 nM T68876 C1JC7K 44307264 Ki = 2500 nM T68876 CX8AL2 56945410 IC50 = 81300 nM T68876 D03NDD 9935648 Ki = 8900 nM T68876 D09VYB 6420161 IC50 = 4000 nM T70680 D02EYG 10096344 IC50 > 100000 nM T70680 D0PW7C 51039 IC50 = 120000 nM T70680 D0X9ZC 47965 Ki = 8620 nM T70680 D0HG2S 86294663 IC50 = 720 nM T70680 D0Z9CC 148200 IC50 = 6600 nM T70680 C49KQP 72740 IC50 = 6500 nM T70680 CM47KI 5351344 IC50 = 16390 nM T70680 CV5X8A 10224181 IC50 = 18000 nM T70680 CI28JY 10457775 IC50 > 200000 nM T70680 CJM90S 11259332 IC50 = 59000 nM T70680 CD19GL 15740213 IC50 = 2300 nM T70680 CHR2P1 25183768 IC50 = 6000 nM T70680 CZL23E 86271138 IC50 = 500 nM T70680 C6CT7S 91099236 IC50 = 1100 nM T70680 CM59EQ 118917669 IC50 = 3300 nM T70680 C6J8YF 118917671 IC50 = 3400 nM T70680 CHB79F 122232270 IC50 = 8300 nM T70680 C7P0MU 155541607 IC50 = 1100 nM T70680 CUCN87 155561820 IC50 = 2800 nM T70680 CRK46A 155565873 IC50 = 1300 nM T70680 D0W4WF 100801 IC50 = 22700 nM T47885 D03ZBT 11626560 IC50 > 10000 nM T47885 D05PZB 135398495 IC50 = 10 nM T47885 D0E3TC 44259 IC50 = 3.6 nM T47885 D03BNU 59604787 IC50 > 10000 nM T47885 D0T3ME 156422 IC50 > 30000 nM T47885 CJ17AM 4877 IC50 = 900 nM T47885 C1EB0M 461195 IC50 = 3100 nM T47885 CACS26 11561968 Ki > 2000 nM T47885 CU0E8O 11690457 Ki > 2000 nM T47885 C9TU1O 16046126 IC50 > 1000 nM T47885 CZF23I 16124479 IC50 = 501.19 nM T47885 CW38QS 25020248 IC50 = 764 nM T47885 CY6I9E 25020250 IC50 = 0.6 nM T47885 CSI54O 25020305 IC50 = 382 nM T47885 C4SV6O 25020308 IC50 = 2 nM T47885 C9OV7I 45258277 IC50 = 28.3 nM T47885 C5WC9K 46871765 IC50 = 650 nM T47885 CVJ4K0 46899547 IC50 > 10000 nM T47885 C2B8IC 46899551 IC50 = 1000 nM T47885 CY3M0L 46899552 IC50 = 4 nM T47885 CVW05P 46899553 IC50 < 1 nM T47885 CV3MG5 46899554 IC50 < 1 nM T47885 CVKT97 46899556 IC50 = 2 nM T47885 CQ58JP 46899557 IC50 = 68 nM T47885 CB4AQ6 46899558 EC50 = 679 nM T47885 CQP5M0 46899718 EC50 = 831 nM T47885 CGU71M 46899719 IC50 = 14 nM T47885 C7IGC8 46899720 IC50 = 25 nM T47885 CZSJ05 46899721 IC50 = 46 nM T47885 CYQL28 46899722 IC50 = 55 nM T47885 CO3SN0 46899723 IC50 > 1000 nM T47885 C7A0LO 46899899 IC50 = 6 nM T47885 C7NSA9 46899901 IC50 = 0.4 nM T47885 C85JKU 46899902 IC50 = 78 nM T47885 CO69NH 46899903 IC50 = 3 nM T47885 CDVN91 46899904 EC50 = 342 nM T47885 C9XET2 46899905 EC50 = 568 nM T47885 CA7G1P 46900065 IC50 = 474 nM T47885 CV0W4N 46900066 IC50 = 2 nM T47885 C42ENY 46900067 IC50 = 454 nM T47885 CZA36B 46900069 IC50 > 1000 nM T47885 CUCH62 46900230 IC50 = 1 nM T47885 C5KF7A 46900231 IC50 = 5 nM T47885 CQ0OI1 46900232 IC50 = 204 nM T47885 C3APD1 46900233 IC50 = 20 nM T47885 C8AYI7 46900234 IC50 = 3 nM T47885 CNFP04 46900235 IC50 = 35 nM T47885 CM1B5E 46900385 IC50 = 4 nM T47885 C81CHW 46900386 IC50 = 3 nM T47885 CAN59P 46900387 IC50 = 3 nM T47885 CN5UR6 46900388 IC50 = 228 nM T47885 CHV6Y2 46900714 IC50 = 12 nM T47885 C31DWK 46900715 IC50 = 695 nM T47885 CY4CV5 46900716 IC50 = 191 nM T47885 CZF70T 46900888 IC50 = 262 nM T47885 CGQ37D 46900889 IC50 = 43 nM T47885 C30OKI 46900891 IC50 = 96 nM T47885 CW78AO 46901053 IC50 = 2 nM T47885 CLW17F 46901056 IC50 = 1 nM T47885 CYPI85 46901211 IC50 = 35 nM T47885 C7MOX5 46901212 IC50 = 1 nM T47885 CA93TO 46901384 IC50 = 1 nM T47885 CU6DN3 46901385 IC50 = 1 nM T47885 CMSE81 46901542 IC50 = 1 nM T47885 CPR3W7 46901543 IC50 = 1 nM T47885 CH8B7K 46901544 IC50 = 1 nM T47885 CWH27M 46901545 EC50 = 202 nM T47885 CQW7I6 46901546 IC50 = 4 nM T47885 CXE9K0 46901547 EC50 = 66 nM T47885 CVM72U 46901548 EC50 = 378 nM T47885 CL4Z9A 46901712 IC50 = 8 nM T47885 CSV5B9 46901859 IC50 = 321 nM T47885 C7YJ2X 46901862 IC50 = 59 nM T47885 CF1AO7 46902013 IC50 < 1 nM T47885 CMS28B 49850059 IC50 = 5.5 nM T47885 CIJ0S7 49864239 IC50 = 19 nM T47885 CCL6T7 49870878 IC50 = 10000 nM T47885 C0MNT5 51346849 IC50 = 3.7 nM T47885 CPA4G0 51346850 IC50 = 9 nM T47885 CL47XT 53317515 IC50 = 111 nM T47885 C53ZSP 53317611 IC50 = 1000 nM T47885 CQ1A7V 53317614 EC50 = 570 nM T47885 CHZ38N 53317615 IC50 = 430 nM T47885 CQ0E5B 53317616 IC50 = 2300 nM T47885 C5OQG1 53320109 IC50 = 124 nM T47885 CSH59W 53320215 IC50 = 280 nM T47885 CL74FI 53320223 IC50 = 6900 nM T47885 CX9P1J 53320224 IC50 = 95 nM T47885 CH8T1Z 53321415 IC50 = 74.9 nM T47885 C8GZ9A 53321416 IC50 = 193 nM T47885 CYB87M 53321529 IC50 = 2500 nM T47885 C05BRF 53321599 IC50 = 87 nM T47885 C8IZF0 53322862 IC50 = 430 nM T47885 C8EJY2 53322863 IC50 = 980 nM T47885 CSDB56 53322873 IC50 = 19 nM T47885 CO5G0L 53324184 IC50 = 390 nM T47885 CGLT40 53324193 IC50 = 200 nM T47885 CZ82ON 53324194 IC50 = 140 nM T47885 CET76D 53324195 IC50 = 2000 nM T47885 CK6PB8 53324196 IC50 = 100 nM T47885 CS5HZ8 53324197 IC50 = 6000 nM T47885 C5LRH2 53325494 IC50 = 1600 nM T47885 CU8V1Y 53325495 IC50 = 1100 nM T47885 CIL5W0 53325496 IC50 = 220 nM T47885 CV0W8P 53325617 IC50 = 130 nM T47885 CJ9U3Q 53326662 IC50 = 750 nM T47885 CLSD56 53326758 IC50 = 200 nM T47885 C3LA0E 53326759 IC50 = 49 nM T47885 CD4H3S 53354074 Ki = 2420 nM T47885 C8NA4L 53384644 IC50 > 30000 nM T47885 C1MR8Q 60097495 IC50 > 1000 nM T47885 CV63UL 67240318 IC50 > 10000 nM T47885 C0ZXY3 86693116 Ki = 14 nM T47885 CBJ1P2 86693157 Ki = 25 nM T47885 CMY4D7 86693162 Ki = 4.9 nM T47885 CU78DC 86693540 Ki < 0.2 nM T47885 CT04ER 89754780 Ki < 0.2 nM T47885 CDEW02 89755037 Ki = 4.2 nM T47885 C6Z7ID 89759863 Ki = 5.9 nM T47885 CH75AV 89759865 Ki = 0.9 nM T47885 C4X7SD 122192466 IC50 > 10000 nM T47885 C6MZL2 134145793 Ki < 0.2 nM T47885 CQDC40 134151887 Ki = 65 nM T47885 CCH37I 134163557 Ki < 0.2 nM T47885 C2MD1Q 155513187 IC50 > 10000 nM T47885 CJP09I 155520168 Ki = 3.6 nM T47885 CS29GT 155528718 Ki = 44 nM T47885 C0FAD1 155540387 Ki < 0.2 nM T47885 CLA0I9 155552645 Ki = 62 nM T47885 D00JGL 6419753 IC50 = 9100 nM T47885 D02XHC 448912 IC50 > 100000 nM T47885 D08JPU 3501 IC50 = 27 nM T47885 D0F2SA 46901383 IC50 = 1 nM T47885 D0GT8N 5154691 IC50 = 250 nM T47885 D0H6ZP 16654987 IC50 = 1000 nM T47885 D0MC3K 755673 IC50 = 182 nM T47885 D0U3NI 53246941 IC50 = 35 nM T50970 D0I0EG 44093 Ki > 10000 nM T50970 D09JES 6324648 IC50 = 1500 nM T50970 D0N4IV 10718956 IC50 > 1000 nM T50970 D02DLE 132968 IC50 = 410 nM T50970 D08GQK 9951814 IC50 = 1300 nM T50970 D0K9YR 9810328 IC50 = 70 nM T50970 D0T2IQ 443600 IC50 = 4000 nM T50970 CO58XD 5311161 IC50 > 100000 nM T50970 CLVN34 5496618 IC50 = 11 nM T50970 CK28XO 9800935 IC50 = 1500 nM T50970 C32XZY 9804685 IC50 = 239.88 nM T50970 CMIP58 9806479 Ki = 10.8 nM T50970 C8J5NE 9820460 IC50 = 1300 nM T50970 CBD5W8 9826127 IC50 = 170 nM T50970 CYV4Z5 9863167 IC50 = 22 nM T50970 C38BVX 9870100 IC50 > 1000 nM T50970 CA76MF 9906947 IC50 = 40 nM T50970 C8X7NJ 9912484 IC50 = 77 nM T50970 CT6KI1 9914454 IC50 = 150 nM T50970 COH8P4 9949799 IC50 > 3000 nM T50970 CVG0O2 9959014 IC50 > 1000 nM T50970 CI2HX5 9969592 IC50 > 3000 nM T50970 C1FM2C 9979153 IC50 = 120 nM T50970 CLQ6Z2 9982912 Ki = 18 nM T50970 C4TZ3C 10014792 IC50 = 190 nM T50970 C98HBI 10028014 IC50 = 4800 nM T50970 CD1J7K 10047910 IC50 = 2000 nM T50970 C83QTK 10050525 IC50 = 37000 nM T50970 CN85LI 10059732 IC50 = 6500 nM T50970 CRBW72 10088334 IC50 = 620 nM T50970 CCR3U8 10093695 IC50 >> 100000 nM T50970 C6NDV0 10132004 IC50 > 3000 nM T50970 CG0DW7 10141595 IC50 = 6.9 nM T50970 CCS45J 10160340 Ki = 22 nM T50970 CZ12NB 10163252 Ki = 31 nM T50970 C3XA7F 10204512 Ki = 35 nM T50970 C5ME3I 10226317 IC50 = 220 nM T50970 C8XWL1 10236332 IC50 = 3 nM T50970 C9NX1V 10330146 IC50 = 3000 nM T50970 C3TFH8 10330979 IC50 = 6.8 nM T50970 CDJ68E 10338615 IC50 = 24000 nM T50970 CG5FK7 10342348 IC50 = 109000 nM T50970 CAH5D0 10344688 IC50 = 61000 nM T50970 CH1A4X 10344880 IC50 = 30 nM T50970 CXW6K8 10376620 IC50 = 0.01 nM T50970 CPK12V 10381623 IC50 = 1700 nM T50970 CX2D0B 10389893 IC50 = 11 nM T50970 CEI64K 10426451 IC50 = 150 nM T50970 CU8FG9 10432455 IC50 >> 100000 nM T50970 CK31SN 10432581 IC50 >> 100000 nM T50970 C2T6YQ 10455810 Ki = 10 nM T50970 CVK75H 10457828 IC50 = 48000 nM T50970 CX38EB 10467565 IC50 > 10000 nM T50970 C9XC8Y 10493383 IC50 > 100000 nM T50970 CTPC82 10501144 IC50 = 110 nM T50970 COZR84 10505477 IC50 = 28 nM T50970 C87HBU 10518365 IC50 = 240 nM T50970 CM1CJ3 10528823 IC50 = 110 nM T50970 C02VDP 10598769 IC50 = 4300 nM T50970 CG0AN8 10601571 IC50 = 8 nM T50970 CG32FM 10613145 IC50 > 100000 nM T50970 C5VGI8 10622593 IC50 = 51 nM T50970 CKDT82 10623498 IC50 > 4000 nM T50970 C7UH9R 10647129 IC50 = 56 nM T50970 CNJ2K9 10647364 IC50 = 130 nM T50970 C02PTU 10648112 IC50 = 34 nM T50970 CW7GR6 10648756 IC50 = 28 nM T50970 CJU8E7 10650987 IC50 = 6.4 nM T50970 CI19VE 10669956 IC50 = 310 nM T50970 CA14CE 10691661 IC50 = 140 nM T50970 C4Z0CX 10694200 IC50 = 150 nM T50970 C82VZE 10696749 IC50 = 43 nM T50970 CSJC70 10715413 IC50 = 250 nM T50970 CZC4M7 10719503 IC50 = 33 nM T50970 CI4SQ2 10732349 IC50 > 10000 nM T50970 C6IB1M 10740493 IC50 = 400 nM T50970 CZAO16 10744617 IC50 = 13 nM T50970 CVA35S 10763731 IC50 = 230 nM T50970 CGE6W5 10764686 IC50 = 110 nM T50970 C57SVI 10766810 IC50 = 53 nM T50970 CX34MD 10768671 IC50 = 82 nM T50970 CLAP90 10785969 IC50 > 1000 nM T50970 CM74LH 10789594 IC50 > 1000 nM T50970 C1UF0K 10791459 IC50 = 25 nM T50970 C3HP5C 10813470 IC50 = 30 nM T50970 CYI19A 10814639 IC50 = 160 nM T50970 CJP19Q 10829413 IC50 = 170 nM T50970 C6B4OW 10834551 IC50 = 510 nM T50970 C3UCL2 10854279 IC50 = 450000 nM T50970 C43HFO 11058931 Ki = 250 nM T50970 CBGX91 11069565 Ki = 1140 nM T50970 CN35IX 11133314 Ki = 290 nM T50970 CC57LQ 11144312 Ki = 1240 nM T50970 CC0MU7 11192220 IC50 = 49.7 nM T50970 CB6Y8N 11505649 IC50 = 39 nM T50970 CE3HA6 11556698 Ki = 14 nM T50970 C7J2OZ 11732301 Ki = 680 nM T50970 C9WK5G 11754555 IC50 = 14 nM T50970 CC2D1U 11761637 Ki = 190 nM T50970 C4ST6H 11797221 IC50 = 520 nM T50970 CJ4VL3 11797382 IC50 > 1000 nM T50970 C0HJ8U 11811641 Ki = 26 nM T50970 C9SJ5L 12068597 IC50 = 650 nM T50970 CF48EI 12068598 IC50 = 850 nM T50970 C7N9MK 12972252 IC50 = 55.98 nM T50970 C3H7JQ 12972253 IC50 = 23.99 nM T50970 C1WE5B 12972254 IC50 = 27 nM T50970 C60EGV 12986821 IC50 = 64 nM T50970 C6TE9U 15411504 IC50 = 1400 nM T50970 C2RDC7 15411506 IC50 = 2600 nM T50970 C5X9MA 15411507 IC50 = 4300 nM T50970 CY71VF 15518148 Ki = 110 nM T50970 C78MDG 15518149 Ki = 28 nM T50970 C7XBS4 15518150 Ki = 90 nM T50970 CV6R0W 15983962 IC50 = 440 nM T50970 C6CU8A 22144624 IC50 = 740 nM T50970 C8RTS3 22144657 IC50 = 390 nM T50970 CA47XT 22144662 IC50 = 210 nM T50970 C2TM8R 22144668 IC50 = 120 nM T50970 C6VJE4 22144671 IC50 = 5900 nM T50970 C5SBD3 22144690 IC50 = 1200 nM T50970 CMD94W 22732542 Ki = 47 nM T50970 CC0O7V 22732546 Ki = 370 nM T50970 CAV67F 22732548 Ki = 210 nM T50970 CTQW09 22732549 Ki = 90 nM T50970 CC1Y0T 22732559 Ki = 100 nM T50970 C0OIV8 22732571 Ki = 79 nM T50970 CZ0S8U 22732575 Ki = 300 nM T50970 CV8I0J 22732589 Ki = 760 nM T50970 CI4MO6 22857947 IC50 = 90 nM T50970 C20ZDR 22857948 IC50 = 50 nM T50970 C01RQG 22857961 IC50 = 60 nM T50970 CR5E6J 22857963 IC50 = 190 nM T50970 CR5C2Z 22857964 IC50 = 120 nM T50970 CYQB03 22859207 IC50 = 12000 nM T50970 CNUA49 23573383 IC50 = 300 nM T50970 CZEQ13 23573393 IC50 = 860 nM T50970 C0IHB9 23573396 IC50 = 6400 nM T50970 CI5P9O 23573398 IC50 = 2300 nM T50970 C7VC5L 23573406 IC50 = 2200 nM T50970 CO6S2I 23573408 IC50 = 3000 nM T50970 CCR10T 23573409 IC50 = 5100 nM T50970 CU30NJ 23573412 IC50 = 170 nM T50970 C9CX2M 23573445 IC50 = 200 nM T50970 C3U9WN 23573446 IC50 = 220 nM T50970 C2FB4Z 24776318 Ki = 220 nM T50970 CC4L6K 24776323 Ki = 100 nM T50970 COTD36 24776324 Ki = 200 nM T50970 CCA0K6 24776325 Ki = 780 nM T50970 CX6H9U 24776326 Ki = 580 nM T50970 CR51QK 24776327 Ki = 110 nM T50970 C8RW9V 24776328 Ki = 135 nM T50970 C07NOG 24776329 Ki = 920 nM T50970 CNCT96 24776330 Ki = 190 nM T50970 CNG1L3 44266455 IC50 = 110 nM T50970 C5Y8EG 44266465 IC50 = 1400 nM T50970 C41APY 44266469 IC50 = 93 nM T50970 C49ZRD 44266477 IC50 = 160 nM T50970 C4VB5X 44266479 IC50 > 1000 nM T50970 CGO98H 44266483 IC50 = 23 nM T50970 C8R9ES 44266484 IC50 = 280 nM T50970 CI3S2Y 44266520 IC50 = 5000 nM T50970 C7GOP6 44266525 IC50 = 17 nM T50970 C4VGW3 44266547 IC50 = 1100 nM T50970 CI5M9G 44266561 IC50 = 390 nM T50970 CD83CF 44266576 IC50 > 1000 nM T50970 C0DUK2 44266601 IC50 > 1000 nM T50970 CN7DR4 44275416 IC50 = 60000 nM T50970 C6I3TP 44275459 IC50 = 50000 nM T50970 C0D1BU 44275460 IC50 = 4300 nM T50970 CBW4U8 44275461 IC50 = 12000 nM T50970 CE48ZG 44275545 IC50 = 25000 nM T50970 CR78JL 44275546 IC50 = 7000 nM T50970 C1XW8V 44275712 IC50 = 20000 nM T50970 CMH8D4 44275713 IC50 = 30000 nM T50970 C6OJV1 44275764 IC50 > 100000 nM T50970 CH06AM 44275765 IC50 = 10000 nM T50970 C7WDL8 44275775 IC50 = 20000 nM T50970 CYN0C4 44275794 IC50 = 5000 nM T50970 C54UHQ 44275795 IC50 > 100000 nM T50970 C7GH6B 44275869 IC50 = 6000 nM T50970 CDAN01 44275870 IC50 = 20000 nM T50970 CPNY12 44275871 IC50 > 100000 nM T50970 CFQ1A9 44275872 IC50 = 20000 nM T50970 CMND16 44275873 IC50 = 400 nM T50970 CSFD75 44275911 IC50 = 4000 nM T50970 CER04J 44275916 IC50 = 80000 nM T50970 C1S6PA 44275933 IC50 = 30000 nM T50970 CNFQ10 44275934 IC50 = 5800 nM T50970 C32HTK 44275937 IC50 = 80000 nM T50970 C4MR2S 44275948 IC50 = 8000 nM T50970 C9IF0V 44283438 Ki = 4150 nM T50970 C6BIS9 44283450 Ki = 900 nM T50970 CS62BV 44283511 Ki = 1560 nM T50970 C9EVM2 44283523 Ki = 300 nM T50970 CX5YP3 44283557 Ki = 980 nM T50970 CTF9X0 44283601 Ki = 600 nM T50970 CS4UN9 44283652 Ki = 670 nM T50970 C98LAG 44283720 Ki > 10000 nM T50970 C1XJ0W 44285058 IC50 = 230 nM T50970 CHG51O 44285096 IC50 = 76 nM T50970 CYT67M 44285121 IC50 = 111 nM T50970 CFL9Y2 44285271 IC50 = 590 nM T50970 C9CQ3N 44289124 IC50 > 1000 nM T50970 CX3BN8 44289125 IC50 > 10000 nM T50970 C0EP2V 44289135 IC50 > 10000 nM T50970 CB85IS 44289136 IC50 > 10000 nM T50970 CI0B1Q 44289330 IC50 = 160 nM T50970 CJ56BX 44289331 IC50 = 250 nM T50970 C7DN3X 44289332 IC50 = 550 nM T50970 C1SBC5 44289366 IC50 = 600 nM T50970 CA53RN 44289649 IC50 = 420 nM T50970 C1XS6T 44292842 IC50 = 15500 nM T50970 C7H5MA 44293049 IC50 = 500 nM T50970 CY3QP6 44293117 IC50 = 1200 nM T50970 CQ34JK 44293118 IC50 = 1300 nM T50970 CLGY89 44293119 IC50 = 4400 nM T50970 C0W5HQ 44293135 IC50 = 1200 nM T50970 C6MOD4 44293143 IC50 = 1200 nM T50970 C9ZEI7 44293144 IC50 = 250 nM T50970 CIR59L 44293161 IC50 = 360 nM T50970 CJ67PU 44293396 IC50 = 2700 nM T50970 CVS3W4 44293558 IC50 = 17700 nM T50970 CG1RQ2 44293559 IC50 = 8950 nM T50970 CFVJ06 44293606 IC50 = 720 nM T50970 C5Y7EG 44293607 IC50 = 700 nM T50970 CB3T6I 44293608 IC50 = 280 nM T50970 CNGY03 44294639 IC50 >> 100000 nM T50970 CVN1E0 44301373 IC50 >> 100000 nM T50970 C4T6ND 44301375 IC50 = 100000 nM T50970 CO9V4C 44301525 IC50 >> 100000 nM T50970 C2WDU4 44301530 IC50 = 31000 nM T50970 CK8O7F 44301550 IC50 = 100000 nM T50970 CR4I0U 44301760 IC50 = 30000 nM T50970 CTD2M7 44301771 IC50 >> 100000 nM T50970 CLC74B 44301772 IC50 = 47000 nM T50970 CS69YV 44301788 IC50 >> 100000 nM T50970 CS6CE3 44303040 Ki = 1460 nM T50970 CR4L1U 44303101 Ki = 140 nM T50970 CR1M7T 44303110 Ki = 10 nM T50970 C2CL3S 44303111 Ki = 100 nM T50970 C6TU7R 44303134 Ki = 560 nM T50970 CW39HV 44303996 IC50 = 210 nM T50970 C70WGD 44303998 IC50 = 200 nM T50970 C6IWR5 44304016 IC50 = 510 nM T50970 C7P5VN 44304017 IC50 = 40 nM T50970 CC93WS 44304019 IC50 = 140 nM T50970 CJ7K8E 44304063 IC50 = 11 nM T50970 CSU1Y8 44304080 IC50 = 19 nM T50970 C8OK5H 44304173 IC50 = 280 nM T50970 CC25KQ 44304321 IC50 = 54 nM T50970 CZ2P1Y 44304467 IC50 = 240 nM T50970 C3FP5R 44304470 IC50 = 170 nM T50970 C6PJW8 44307469 IC50 = 860 nM T50970 CQP9Y0 44307536 IC50 = 1300 nM T50970 CW4O1K 44307550 IC50 > 50000 nM T50970 C1EB5K 44307551 IC50 = 2400 nM T50970 CO3Z7N 44307560 IC50 = 1400 nM T50970 CPYB80 44307561 IC50 = 10000 nM T50970 CQ8O7X 44307680 IC50 > 10000 nM T50970 CD3XM7 44307681 IC50 > 10000 nM T50970 CIB2W1 44307691 IC50 = 24000 nM T50970 C0AIW4 44307702 IC50 > 50000 nM T50970 C3ZA8T 44307703 IC50 > 50000 nM T50970 CFK69H 44307709 IC50 > 10000 nM T50970 CO9QR7 44307715 IC50 = 980 nM T50970 CK0Y4R 44307732 IC50 = 1500 nM T50970 CX47FJ 44307743 IC50 = 10000 nM T50970 CMWO72 44307759 IC50 = 500 nM T50970 CQ2Y7F 44307822 IC50 = 4.8 nM T50970 CDV23J 44307823 IC50 = 0.25 nM T50970 C0CL9N 44307977 IC50 = 0.2 nM T50970 CS8F6B 44307978 IC50 = 1.2 nM T50970 C2KYL0 44307980 IC50 = 10000 nM T50970 CJX52D 44308003 IC50 = 3000 nM T50970 CH9VM4 44308023 IC50 = 150 nM T50970 CG0R2L 44334175 IC50 = 82 nM T50970 CQ0R7D 44334182 IC50 = 130 nM T50970 CB2M4V 44334195 IC50 = 9.795 nM T50970 CYFO71 44334230 IC50 = 23.01 nM T50970 C87VIN 44334236 IC50 = 699.84 nM T50970 C3QC8M 44334243 IC50 = 41.02 nM T50970 C7H2VO 44334267 IC50 = 9.5 nM T50970 CH6AT0 44334306 IC50 = 77 nM T50970 CHN39B 44334329 IC50 = 43 nM T50970 CI6A0B 44334333 IC50 = 120 nM T50970 C0B2TE 44334343 IC50 = 39 nM T50970 CK4C9L 44334454 IC50 = 98 nM T50970 C2QLC5 44334502 IC50 = 54.95 nM T50970 C08EWN 44334555 IC50 = 48.98 nM T50970 CCXW90 44348629 IC50 = 650 nM T50970 C50OJI 44348671 IC50 = 560 nM T50970 CQ2DK4 44348758 IC50 = 180 nM T50970 CEI42C 44348865 IC50 = 990 nM T50970 CSCJ68 44348873 IC50 = 150 nM T50970 CV1P2C 44348879 IC50 = 220 nM T50970 C9G1NE 44348880 IC50 = 300 nM T50970 C8C7ZY 44348883 IC50 = 350 nM T50970 CY3B4A 44348890 IC50 = 130 nM T50970 CNY56R 44348897 IC50 = 490 nM T50970 C5WIK0 44348910 IC50 = 320 nM T50970 C0JSI1 44348920 IC50 = 810 nM T50970 CCJ17Y 44348933 IC50 = 650 nM T50970 CKOM58 44348947 IC50 = 370 nM T50970 C03FRV 44364333 IC50 = 2.6 nM T50970 C48CLK 44364365 IC50 = 29 nM T50970 CE9BJ1 44364366 IC50 = 19 nM T50970 CEX8B4 44364381 IC50 = 24 nM T50970 C3TUB9 44364386 IC50 = 35 nM T50970 C1XKN9 44364400 IC50 = 22 nM T50970 C90ZOL 44364412 IC50 = 23 nM T50970 CQ2GI8 44364476 IC50 = 14 nM T50970 C8PVK9 44364478 IC50 = 96 nM T50970 CWJB41 44364533 IC50 = 13 nM T50970 CYZN06 44364534 IC50 = 40 nM T50970 C18MAW 44364547 IC50 = 97 nM T50970 CAOD34 44364643 IC50 = 6 nM T50970 CH6L5O 44364676 IC50 = 65 nM T50970 C0CX5T 44371314 IC50 = 7700 nM T50970 CYF27Z 44371340 IC50 = 5200 nM T50970 CW21NL 44371361 IC50 = 5400 nM T50970 CHP89K 44371476 IC50 = 7800 nM T50970 CFG1H2 44371519 IC50 = 5200 nM T50970 CD19SU 44371685 IC50 = 6500 nM T50970 C8MW0N 44371700 IC50 = 6500 nM T50970 CTFS09 44384017 IC50 > 10000 nM T50970 CF2I3D 44388021 IC50 = 10890 nM T50970 C1FRV0 44400757 IC50 = 61.3 nM T50970 CK79BM 44400838 IC50 = 16 nM T50970 C8J4XB 44401169 IC50 = 72.9 nM T50970 CR9MN8 44403588 IC50 = 130 nM T50970 CPD5J8 44403604 IC50 > 10000 nM T50970 CSDC96 44403610 IC50 > 10000 nM T50970 CTMH76 44403613 IC50 > 10000 nM T50970 C9UQ3X 44403614 IC50 = 150 nM T50970 C2X6GT 44403615 IC50 = 66 nM T50970 CMQ0A9 44403616 IC50 = 120 nM T50970 CE0VK1 44403624 IC50 = 660 nM T50970 C8XV6R 44403631 IC50 = 6700 nM T50970 CWR0Y2 44403632 IC50 = 7000 nM T50970 CO9BW0 44403637 IC50 = 7400 nM T50970 CG5QO6 44403638 IC50 > 10000 nM T50970 CAE21M 44413731 IC50 > 3000 nM T50970 C90RTX 44413815 IC50 > 3000 nM T50970 CIO42C 44460248 IC50 = 5050 nM T50970 CA1YC9 44626604 Ki = 26 nM T50970 CK6S5H 44626708 Ki = 8 nM T50970 C0EJ1F 44626709 Ki = 240 nM T50970 CZR23J 44626710 Ki = 7.7 nM T50970 CQB06H 44626711 Ki = 275 nM T50970 C17IGS 44627959 Ki = 910 nM T50970 CM1DL3 44627960 Ki = 2100 nM T50970 CNZ8L0 44628063 Ki > 5000 nM T50970 CRU86P 44628064 Ki > 10000 nM T50970 CS5BG9 44628065 Ki > 10000 nM T50970 C65RAJ 45102601 IC50 = 79.43 nM T50970 C03HVM 45267758 IC50 > 10000 nM T50970 CJ73YP 45267767 IC50 > 10000 nM T50970 CG80EY 45269496 IC50 > 10000 nM T50970 CT15VE 45270333 IC50 > 10000 nM T50970 C48XKY 45272068 IC50 > 10000 nM T50970 CX4DS1 45273826 IC50 = 2420 nM T50970 CTOA14 45485236 Ki = 14 nM T50970 CG7L5T 53824916 IC50 = 54.08 nM T50970 CGH0S7 54589400 IC50 > 100000 nM T50970 CZD09H 56668219 IC50 > 100000 nM T50970 C7HA0D 59902420 IC50 = 650.13 nM T50970 C0Z6TU 71452809 IC50 = 97 nM T50970 C9D6KR 71459988 IC50 = 410 nM T50970 CK0N7F 71460032 IC50 = 4000 nM T50970 C7F0WO 73349980 IC50 = 33000 nM T50970 C1FJ9H 74988248 IC50 = 510.5 nM T50970 CLW2N5 76309557 IC50 = 199.99 nM T50970 CQCL08 76313233 IC50 = 179.89 nM T50970 C4Q1WS 76313234 IC50 = 130.02 nM T50970 CR3ZF7 76313235 IC50 = 810.96 nM T50970 CVUQ30 76313236 IC50 = 19.01 nM T50970 CIBZ65 76313237 IC50 = 97.05 nM T50970 CT3X1F 76313238 IC50 = 139.96 nM T50970 CV8ZD5 76316776 IC50 = 650.13 nM T50970 CWG0N6 76320475 IC50 = 319.89 nM T50970 CQ39YA 76320476 IC50 = 170.22 nM T50970 C6D3QU 76320477 IC50 = 209.89 nM T50970 C3T6MS 76320478 IC50 = 119.95 nM T50970 CNY29P 76324134 IC50 = 489.78 nM T50970 CUY4P8 76327683 IC50 = 410.2 nM T50970 C6RX8C 76327684 IC50 = 39.99 nM T50970 C2NY7L 76331357 IC50 = 561.05 nM T50970 CL3DV7 76331358 IC50 = 11.02 nM T50970 CWA12V 76334941 IC50 = 299.92 nM T50970 CA14PT 76334942 IC50 = 369.83 nM T50970 CAX25C 76334943 IC50 = 10.99 nM T50970 CJ7B1X 76334944 IC50 = 279.9 nM T50970 C54ESG 90668209 IC50 > 31622.78 nM T50970 CX4MK8 90668210 IC50 > 31622.78 nM T50970 CX5MA6 90668211 IC50 > 31622.78 nM T50970 C3YZO5 90668278 IC50 > 31622.78 nM T50970 C6OPV5 118719300 IC50 = 120 nM T50970 C9QKI3 127020966 IC50 > 100000 nM T50970 C9HPG8 137661516 IC50 > 300 nM T50970 CU42CE 155567829 IC50 > 100000 nM T50970 D02BTV 9816867 IC50 > 100000 nM T50970 D04QJY 123982 IC50 = 8 nM T50970 D07APP 131255 IC50 = 12 nM T50970 D08ELY 9838786 IC50 > 50000 nM T50970 D09NAJ 445114 IC50 = 100 nM T50970 D0F8AR 45485268 Ki = 1.2 nM T50970 D0K1MA 9913857 IC50 = 20000 nM T50970 D0N6CD 10565532 IC50 = 78000 nM T50970 D0PB5Q 3132 IC50 = 8 nM T98278 D00JAU 3749 Ki = 0.8 nM T98278 D00NVX 132706 IC50 = 6.9 nM T98278 D04JEE 4946 EC50 > 5011.87 nM T98278 D06UDG 60846 IC50 = 2.7 nM T98278 D0D5SQ 2541 IC50 = 0.69 nM T98278 D0G6SE 172198 Ki = 0.16 nM T98278 D0K0AT 6324663 Ki = 0.17 nM T98278 D0M7TO 60919 IC50 = 32 nM T98278 D0N6RF 65999 IC50 = 0.49 nM T98278 D0T7US 5281037 IC50 = 7.3 nM T98278 D02BBC 6918269 IC50 = 6 nM T98278 D0LI1C 44469321 IC50 > 30000 nM T98278 D0O0JP 9937291 IC50 = 39 nM T98278 D0X2XF 177336 Ki > 10000 nM T98278 D0YS1U 10257882 Ki = 0.8 nM T98278 D00UBK 9851889 IC50 = 1.7 nM T98278 D04AOA 9954408 IC50 = 12 nM T98278 D05UQD 656629 Ki > 10000 nM T98278 D06TZT 132840 Ki = 24 nM T98278 D07LEW 131590 Ki = 29 nM T98278 D0A8HL 3081289 IC50 = 6 nM T98278 D0A9BX 133031 IC50 = 0.2 nM T98278 D0B3CY 121879 IC50 = 3600 nM T98278 D0B5PU 9843631 Ki > 0.0001 nM T98278 D0E3XG 72168 Ki = 1.995 nM T98278 D0F5VB 5311345 Ki = 12 nM T98278 D0GS7N 183134 IC50 = 2.7 nM T98278 D0J2NB 23703120 IC50 = 0.4 nM T98278 D0N5CT 132404 Ki = 20 nM T98278 D0RG2P 9931685 IC50 = 5.6 nM T98278 CN8XG9 156690 Ki > 10 nM T98278 C2J1RE 351037 IC50 > 79000 nM T98278 C1ICH6 1315061 IC50 = 2089.3 nM T98278 C6IPC5 2121575 IC50 = 2570.4 nM T98278 CA61KC 2121583 IC50 = 199 nM T98278 CYIE52 4803452 IC50 = 2187.76 nM T98278 C20VPT 5249743 Ki = 25 nM T98278 CS1W5V 5284633 IC50 = 300 nM T98278 C08QYK 5311348 IC50 > 100000 nM T98278 CX9FV4 7217852 IC50 > 79000 nM T98278 CR1QE5 7217853 IC50 > 79000 nM T98278 C12BHY 7217856 IC50 > 79000 nM T98278 C86MDE 7217859 IC50 > 79000 nM T98278 C9UBG6 7217861 IC50 > 79000 nM T98278 C3XLA7 7217862 IC50 > 79000 nM T98278 C4Y6JF 7217867 IC50 > 79000 nM T98278 CB8NT2 7217870 IC50 > 79000 nM T98278 CT6F3C 7217876 IC50 > 79000 nM T98278 C8PK9D 7217878 IC50 > 79000 nM T98278 CYX8F6 7217879 IC50 > 79000 nM T98278 CH3I6U 7217884 IC50 > 79000 nM T98278 CI92NG 7217887 IC50 > 79000 nM T98278 C17GSL 7217891 IC50 > 79000 nM T98278 C1W3XE 7217912 IC50 > 79000 nM T98278 C8RWT6 7217913 IC50 > 79000 nM T98278 CFOJ16 7217916 IC50 > 79000 nM T98278 C5LZ0X 7217919 IC50 > 79000 nM T98278 CNG45O 7217921 IC50 > 79000 nM T98278 C2PQ8W 7217922 IC50 > 79000 nM T98278 CA7EW6 7217938 IC50 > 79000 nM T98278 CK9X8S 7217939 IC50 > 79000 nM T98278 CT89GV 7217942 IC50 > 79000 nM T98278 C07ZXA 7217944 IC50 > 79000 nM T98278 CUA9S4 7217946 IC50 > 79000 nM T98278 C7AMT6 7217947 IC50 > 79000 nM T98278 CCE5T6 7217950 IC50 > 79000 nM T98278 CW2AT7 7218011 IC50 > 79000 nM T98278 CZI91W 9807029 IC50 = 0.3 nM T98278 C35FCP 9810305 IC50 = 1.8 nM T98278 CT13BE 9823146 IC50 = 16 nM T98278 C91GBS 9824568 IC50 = 11 nM T98278 CPT7L5 9826191 Ki = 0.5012 nM T98278 C8TD2L 9826888 Ki = 0.48 nM T98278 C1I6GK 9850811 IC50 = 1 nM T98278 CIWU91 9850834 IC50 = 1.5 nM T98278 CV07NF 9851082 IC50 = 1 nM T98278 C2C4OM 9852384 IC50 = 1.4 nM T98278 CRP84D 9853391 IC50 = 0.2 nM T98278 C0BH3O 9869504 IC50 = 1.2 nM T98278 C19NOU 9870652 IC50 = 4.5 nM T98278 CG7I2Q 9871837 IC50 = 2 nM T98278 CQ4LC2 9872676 Ki = 3710 nM T98278 C6SHG0 9874508 IC50 = 8.1 nM T98278 CEO03B 9889557 IC50 = 17 nM T98278 CV8A6J 9895212 IC50 = 0.05 nM T98278 CD04YO 9895957 IC50 = 6 nM T98278 C2M4BW 9895984 IC50 = 4 nM T98278 CB0A3I 9896251 IC50 = 13 nM T98278 CI4A8R 9915892 IC50 = 4.2 nM T98278 CY9N3R 9918412 IC50 = 0.2 nM T98278 CP45TL 9939191 Ki = 1.7 nM T98278 C65CYH 9940350 IC50 = 0.5 nM T98278 CJF49M 9960721 IC50 = 1.9 nM T98278 CRL65O 9979771 IC50 = 2.4 nM T98278 C78POU 9981102 IC50 = 7.1 nM T98278 C86VWU 9983135 IC50 = 11.1 nM T98278 C9DAJ6 9984181 IC50 = 0.9 nM T98278 C6HQP8 9984303 IC50 = 2.7 nM T98278 CG0ET4 9987414 IC50 = 0.74 nM T98278 CG8CL2 10004489 Ki = 0.66 nM T98278 CPR16C 10004498 Ki = 0.49 nM T98278 CFTL14 10004646 IC50 = 2.3 nM T98278 C0GTJ4 10005741 Ki = 2.1 nM T98278 CYF76W 10005890 IC50 = 3 nM T98278 C7DIK2 10006693 IC50 = 9.9 nM T98278 CO3PR5 10007306 IC50 = 4.8 nM T98278 CK62VT 10007312 IC50 = 3.3 nM T98278 CA47HV 10007362 IC50 = 0.5 nM T98278 C1J7MU 10007528 IC50 = 18.5 nM T98278 C59NJL 10009984 IC50 = 0.45 nM T98278 CE5H3C 10010071 IC50 = 0.38 nM T98278 CEI76X 10010164 IC50 = 17 nM T98278 C62DQJ 10026681 IC50 = 4.2 nM T98278 C0C5FR 10027175 IC50 = 3.4 nM T98278 CR60PM 10028164 Ki = 4.3 nM T98278 CMX71V 10029695 IC50 = 11.1 nM T98278 CY8KS9 10030086 IC50 = 1.7 nM T98278 CS0BA9 10030110 IC50 = 0.6 nM T98278 C7QU3W 10030426 IC50 = 14.6 nM T98278 CCS31D 10032820 IC50 = 0.32 nM T98278 CE9XN3 10032851 IC50 = 0.5 nM T98278 CY62AG 10032877 IC50 = 0.88 nM T98278 CT6M8J 10032988 IC50 = 0.41 nM T98278 CJ3D0B 10033136 IC50 = 1.9 nM T98278 CY1ZL5 10047444 IC50 = 4530 nM T98278 CDH6Y0 10048770 IC50 = 6.6 nM T98278 CHDB84 10049809 IC50 = 4 nM T98278 C0UX2N 10050044 Ki = 1.3 nM T98278 CS2QT0 10052319 IC50 = 54.5 nM T98278 CUP97S 10052399 IC50 = 0.6 nM T98278 CRJ4P0 10053110 IC50 = 3 nM T98278 C3O6GI 10053367 IC50 = 11.1 nM T98278 CQUS95 10053595 IC50 = 5 nM T98278 CC5GW1 10075811 IC50 = 3.4 nM T98278 CJ9T2Q 10076109 IC50 = 260 nM T98278 CXOA48 10076191 IC50 = 6.4 nM T98278 C6FP7N 10077513 IC50 = 21.9 nM T98278 CRS30P 10078475 IC50 = 28 nM T98278 CCM3D8 10078554 IC50 = 4.3 nM T98278 C3KX6E 10078780 IC50 = 0.94 nM T98278 C6YFD0 10078800 IC50 = 16 nM T98278 CNQ97X 10079601 Ki = 0.65 nM T98278 CTZ5D8 10095241 Ki = 4.3 nM T98278 CC2IQ7 10095683 Ki = 14 nM T98278 CLW5B0 10095986 IC50 = 2.6 nM T98278 CS3W7A 10096683 Ki = 3.9 nM T98278 C8DE6W 10098291 IC50 = 35.7 nM T98278 CS73XM 10100951 IC50 = 0.28 nM T98278 CM9N8U 10101351 IC50 = 0.34 nM T98278 CS7A5F 10101606 IC50 = 0.72 nM T98278 C3F0TU 10101608 IC50 = 0.55 nM T98278 CFN78G 10101690 IC50 = 1.4 nM T98278 CAJ86X 10166561 IC50 = 30 nM T98278 CS7K0L 10209324 IC50 = 2 nM T98278 CKX80Y 10254585 IC50 = 1.3 nM T98278 CW17PJ 10254899 Ki = 8.7 nM T98278 C6HV1R 10255888 IC50 = 446 nM T98278 CG1T0D 10256564 IC50 = 8.5 nM T98278 CUK72W 10256602 IC50 = 0.6 nM T98278 CB93EA 10257293 IC50 = 117 nM T98278 C8KAP3 10257584 IC50 = 5.3 nM T98278 C4ZSK2 10259265 IC50 = 14 nM T98278 CU58CL 10259447 IC50 = 0.36 nM T98278 CEYO10 10259468 IC50 = 0.43 nM T98278 CUA9G7 10259525 IC50 = 1.6 nM T98278 CI0WR6 10259841 IC50 = 1.6 nM T98278 C5LC9E 10280531 IC50 = 24 nM T98278 CO9IC8 10322229 Ki = 1 nM T98278 C1QSM9 10323969 IC50 = 16.6 nM T98278 C6V7WG 10324179 IC50 = 15.9 nM T98278 CH21JQ 10324361 IC50 = 10.1 nM T98278 CMX95I 10324657 IC50 = 12.4 nM T98278 CGV5U6 10324870 IC50 = 8 nM T98278 CHJ4G0 10325267 IC50 = 1.2 nM T98278 CHTL80 10325295 IC50 = 47.9 nM T98278 C9P6UA 10325483 IC50 = 4.9 nM T98278 CZ6ML9 10325767 IC50 = 16.9 nM T98278 CJ9H8M 10327309 IC50 < 0.3 nM T98278 CNZ05L 10327728 IC50 = 24 nM T98278 CW7K4Z 10342301 IC50 = 2.8 nM T98278 C4XZO9 10343090 IC50 = 3.5 nM T98278 CAUB84 10344188 Ki = 0.65 nM T98278 CNOX21 10345537 Ki = 2.7 nM T98278 CLIH83 10349897 IC50 = 4.6 nM T98278 CX1A2T 10350123 IC50 = 4.7 nM T98278 C29KUZ 10366402 Ki = 1.1 nM T98278 CWZ9N7 10367792 IC50 = 7.1 nM T98278 C2NBG6 10369479 IC50 = 40.2 nM T98278 CVD5W6 10369701 IC50 = 5.8 nM T98278 CSUH47 10369867 IC50 = 1.5 nM T98278 CTR4A7 10369902 IC50 = 9 nM T98278 CRVA34 10371118 IC50 = 14.3 nM T98278 C6C8UJ 10371295 IC50 = 159 nM T98278 CK24ZW 10372451 IC50 = 0.44 nM T98278 C8PUW5 10372550 IC50 = 2.2 nM T98278 CAU4G3 10372659 IC50 = 0.76 nM T98278 CWAP07 10372810 IC50 = 5.9 nM T98278 CDJ5M3 10373120 IC50 = 0.96 nM T98278 CNW30P 10390188 Ki = 0.29 nM T98278 C8EBV1 10391038 IC50 = 8.5 nM T98278 C6G3FE 10391950 IC50 = 41.7 nM T98278 C5E8WI 10392378 IC50 = 1.2 nM T98278 C70JVE 10393016 Ki = 10 nM T98278 C9VR4Z 10393086 IC50 = 17.6 nM T98278 C5KEW8 10394727 IC50 = 6 nM T98278 CA07JQ 10394859 IC50 = 6.1 nM T98278 C2WXC5 10395076 IC50 = 0.14 nM T98278 CQB57G 10395335 IC50 = 0.43 nM T98278 C7KY3L 10408794 IC50 = 3.467 nM T98278 C9MRQ6 10414273 IC50 = 8.3 nM T98278 C1XST2 10414338 IC50 = 0.7 nM T98278 C42BDV 10414470 IC50 = 1.4 nM T98278 C5KSE6 10415119 IC50 = 14.5 nM T98278 CB0ZK1 10417195 IC50 = 15 nM T98278 C8QY7E 10417321 IC50 = 3.4 nM T98278 C6FSG7 10439715 IC50 = 0.64 nM T98278 C41IQS 10439819 IC50 = 0.4 nM T98278 CO1V5L 10439837 IC50 = 1 nM T98278 C9GM1L 10439858 IC50 = 8.8 nM T98278 CG1Q7I 10440144 IC50 = 2 nM T98278 C37VCL 10459724 IC50 = 245 nM T98278 C1IL2S 10459992 IC50 = 31 nM T98278 CQ08FG 10460186 IC50 = 23.9 nM T98278 CT61DH 10462573 IC50 = 2.2 nM T98278 C8PCF5 10462598 IC50 = 0.32 nM T98278 CV93HT 10462683 IC50 = 1 nM T98278 CCG2B9 10462933 IC50 = 1.1 nM T98278 CUW9F1 10475382 IC50 = 30 nM T98278 C5IFH8 10478294 IC50 = 4.9 nM T98278 CJ03BC 10478476 IC50 = 44 nM T98278 C7JVR6 10479983 Ki = 0.45 nM T98278 CO83VF 10480064 Ki = 9.6 nM T98278 CT5PQ2 10480309 IC50 = 0.5 nM T98278 CB2QK9 10481196 Ki = 2.7 nM T98278 C1HTM9 10481968 IC50 = 1.4 nM T98278 C8TC5F 10482340 IC50 = 47.8 nM T98278 CL8T2A 10482886 IC50 = 9.8 nM T98278 CQE84K 10483597 IC50 = 4.2 nM T98278 C3XK5L 10504330 Ki = 158 nM T98278 CC8X7L 10507383 Ki = 32 nM T98278 CU1Z3D 10623969 Ki > 10000 nM T98278 CXK68V 10643268 Ki > 10000 nM T98278 CQ42UA 10673314 Ki > 10000 nM T98278 C0GO1E 10674630 Ki = 25 nM T98278 C0IDF4 10695091 Ki > 10000 nM T98278 C1G8FB 10695405 Ki = 398 nM T98278 CZRC03 10697700 Ki = 13 nM T98278 CS2U9K 10697829 Ki = 40 nM T98278 CW90RU 10742620 Ki = 29 nM T98278 C3BYA7 10744859 Ki = 42 nM T98278 CJ7A6K 10763626 IC50 = 9.1 nM T98278 CR2WI1 10764613 Ki = 3162 nM T98278 C5DM4Y 10765881 Ki = 3301 nM T98278 CHP75M 10790260 Ki = 1995 nM T98278 CK4W1Q 10790818 Ki = 381 nM T98278 C5B2HR 10790819 Ki = 402 nM T98278 C9A2FH 10811054 Ki > 10000 nM T98278 C35BIO 10884983 Ki = 80 nM T98278 CV2E4Z 11476710 IC50 = 5.5 nM T98278 CT4KU3 11502835 IC50 = 3 nM T98278 CN4GI8 11561462 IC50 = 60 nM T98278 CVH5U6 11754146 Ki = 0.7 nM T98278 CN5AZ0 11754586 Ki = 12 nM T98278 CN9W0D 11757112 IC50 = 34.6 nM T98278 CJ6D4Q 11757216 IC50 = 198 nM T98278 C0G7ME 11757908 IC50 = 104 nM T98278 CL0X3B 11758329 IC50 = 70 nM T98278 CSQ3P5 11758341 IC50 = 8 nM T98278 CUJ7E0 11758470 IC50 = 17.8 nM T98278 CDGF69 11765177 IC50 = 3.3 nM T98278 CD7E5Q 11765454 IC50 = 1.5 nM T98278 C9I0HX 11765560 IC50 = 0.84 nM T98278 CZ2C1H 11801362 Ki = 32 nM T98278 C9ZEC8 12005825 IC50 > 79000 nM T98278 C1D7HW 12005898 IC50 > 79000 nM T98278 C4K8HT 12005992 IC50 > 79000 nM T98278 CD45PU 14952903 IC50 = 440 nM T98278 CQZ71Y 15222070 IC50 = 2 nM T98278 CG5XH2 15222092 IC50 = 2 nM T98278 CBPL06 15222094 IC50 = 2 nM T98278 CO5V6R 15222101 IC50 = 10 nM T98278 CO71QD 15222103 IC50 = 6 nM T98278 CF57HL 15292111 IC50 = 10 nM T98278 CX75ZV 15292112 IC50 = 12 nM T98278 CG29NO 15292113 IC50 = 0.71 nM T98278 CSK27N 15818746 IC50 = 9 nM T98278 CV40ST 15818748 IC50 = 1 nM T98278 CB78RO 16130452 Ki > 100000 nM T98278 C0A9WY 16194671 IC50 > 79000 nM T98278 C6J4NC 16805942 IC50 > 79000 nM T98278 C21UXH 16832372 IC50 > 79000 nM T98278 C8NGJ0 18004820 IC50 = 21 nM T98278 C9IP8D 18572334 IC50 > 79000 nM T98278 CK2L9R 18572335 IC50 > 79000 nM T98278 CO48HV 18572337 IC50 = 60100 nM T98278 CC70BA 18572338 IC50 > 79000 nM T98278 CMG17E 18572343 IC50 > 79000 nM T98278 CQ3ZV0 18572352 IC50 > 79000 nM T98278 CZ2FW0 18572378 IC50 > 79000 nM T98278 COP52X 18572379 IC50 > 79000 nM T98278 CAJH61 18572382 IC50 > 79000 nM T98278 CNKA87 18572395 IC50 > 79000 nM T98278 CL94NS 18654313 IC50 = 661 nM T98278 CA82PW 19008901 IC50 = 96 nM T98278 CT7ED5 19008935 IC50 = 238 nM T98278 CAG89Z 19102815 IC50 = 150 nM T98278 C8BLT0 19430442 IC50 = 0.28 nM T98278 CVL4G0 19430458 IC50 = 0.74 nM T98278 C60YHR 19430462 IC50 = 0.35 nM T98278 CRC30I 19430475 IC50 = 0.57 nM T98278 CVF5K9 19430479 IC50 = 0.6 nM T98278 CSD1U8 19919870 IC50 = 884 nM T98278 C2KQ7M 19939495 IC50 = 110 nM T98278 CBZ9S7 20081627 IC50 = 1.8 nM T98278 C5FZX8 20747575 IC50 = 8 nM T98278 C0X4NY 21840324 IC50 = 30 nM T98278 CK4H2W 21840429 IC50 = 600 nM T98278 C8JZT4 22574723 IC50 = 1.3 nM T98278 CFP01R 24828743 Ki = 549.54 nM T98278 C0TR3U 25190005 Ki = 5.012 nM T98278 C8TX1U 42281625 IC50 > 79000 nM T98278 CE69MC 44210864 IC50 = 3 nM T98278 C5FDC2 44254496 Ki = 141.25 nM T98278 CR28CF 44264673 IC50 = 22 nM T98278 C5J6NY 44277442 IC50 = 6.9 nM T98278 C4VK6Q 44277443 IC50 = 5.7 nM T98278 CNX92H 44277461 IC50 = 21.4 nM T98278 CE8TQ6 44277549 IC50 = 10.6 nM T98278 CYIF37 44277567 IC50 = 4.4 nM T98278 CM1K2L 44277573 IC50 = 0.9 nM T98278 CK81TH 44277574 IC50 = 5.09 nM T98278 C97IVT 44277593 IC50 = 9.6 nM T98278 CSC65I 44277594 IC50 = 6 nM T98278 C9TP0H 44277677 IC50 = 4 nM T98278 C93WRI 44277871 IC50 = 4.9 nM T98278 C7VM0B 44285157 IC50 = 100 nM T98278 CO2J0U 44285177 IC50 = 20 nM T98278 CH10OD 44285178 IC50 = 3 nM T98278 CGA4L5 44285212 IC50 = 1400 nM T98278 CV3WH8 44285267 IC50 = 0.9 nM T98278 CCF0T1 44285327 IC50 = 8 nM T98278 C8MR7S 44285370 IC50 = 4 nM T98278 CQD25K 44285371 IC50 = 300 nM T98278 C7VY6C 44285372 IC50 = 2 nM T98278 CJSW19 44301981 IC50 = 44 nM T98278 C4MH6O 44311071 IC50 = 1 nM T98278 C04OWQ 44311072 IC50 = 0.1 nM T98278 CVXU13 44311073 IC50 = 0.1 nM T98278 C64VDR 44311074 IC50 = 0.2 nM T98278 C3O6SW 44311182 IC50 = 0.5 nM T98278 CCD7K5 44311183 IC50 = 0.8 nM T98278 CDC7V8 44311184 IC50 = 0.6 nM T98278 CYSE79 44311185 IC50 = 0.3 nM T98278 CFO20B 44311289 IC50 = 0.2 nM T98278 C5FI1X 44311342 IC50 = 10 nM T98278 CHW83V 44311406 IC50 = 20 nM T98278 C37PFG 44311412 IC50 = 0.2 nM T98278 CAK8C2 44311413 IC50 = 0.2 nM T98278 CHJP87 44311414 IC50 = 0.1 nM T98278 C3WZY9 44311415 IC50 = 0.1 nM T98278 COTX54 44311428 IC50 = 10 nM T98278 C8C5HR 44311429 IC50 = 40 nM T98278 CW7V8A 44311434 IC50 = 0.1 nM T98278 CT6A4H 44311435 IC50 = 0.1 nM T98278 C7FH8G 44311436 IC50 = 3 nM T98278 C5P6NM 44311449 IC50 = 10 nM T98278 CWVO75 44311450 IC50 = 10 nM T98278 CL68EO 44311451 IC50 = 2 nM T98278 C3H1MD 44311452 IC50 = 0.5 nM T98278 C3F6SU 44311453 IC50 = 0.4 nM T98278 C6Q0UC 44311454 IC50 = 0.3 nM T98278 C7SD4Z 44311455 IC50 = 0.1 nM T98278 CKT0U8 44311456 IC50 = 0.2 nM T98278 C5HPL4 44311472 IC50 = 100 nM T98278 C23KJT 44311496 IC50 = 8 nM T98278 C9CY1G 44311497 IC50 = 2 nM T98278 CC9Y6E 44311498 IC50 = 3 nM T98278 CL9Z1B 44311499 IC50 = 2 nM T98278 CRF13T 44311537 IC50 = 0.3 nM T98278 CKI10X 44311538 IC50 = 0.8 nM T98278 COI20G 44311543 IC50 = 10 nM T98278 C4FAK2 44311557 IC50 = 0.3 nM T98278 CB41MY 44311558 IC50 = 0.6 nM T98278 C3X1AL 44311567 IC50 = 9 nM T98278 CY7DG6 44311568 IC50 = 20 nM T98278 C1XC8Q 44311569 IC50 = 20 nM T98278 CD4ZM5 44311571 IC50 = 9 nM T98278 C5UBK7 44311580 IC50 = 0.1 nM T98278 CX90KA 44311581 IC50 = 0.2 nM T98278 CT05AS 44311582 IC50 = 0.2 nM T98278 CUAI35 44311583 IC50 = 2 nM T98278 CTP18U 44311584 IC50 = 8 nM T98278 C04GME 44311607 IC50 = 6 nM T98278 C0R6QJ 44311609 IC50 = 30 nM T98278 C5LJ8A 44311616 IC50 = 9 nM T98278 CSH0R1 44311617 IC50 = 0.6 nM T98278 C92KSW 44311618 IC50 = 0.6 nM T98278 CPGV60 44311619 IC50 = 0.4 nM T98278 CSE80D 44311635 IC50 = 0.9 nM T98278 C6CQ3Y 44311636 IC50 = 20 nM T98278 CLT7J0 44311638 IC50 = 30 nM T98278 CXZ1Y2 44311648 IC50 = 2 nM T98278 CX89YT 44311650 IC50 = 6 nM T98278 CU4HB9 44311662 IC50 = 2 nM T98278 C0I8FS 44311663 IC50 = 2 nM T98278 CT1X8Z 44311664 IC50 = 10 nM T98278 CR7Q4V 44311675 IC50 = 0.3 nM T98278 C3X7ZI 44311676 IC50 = 0.1 nM T98278 C8SY2D 44311681 IC50 = 2 nM T98278 C46NML 44311683 IC50 = 0.4 nM T98278 CP7CY2 44311688 IC50 = 10 nM T98278 CJ9A7D 44311715 IC50 = 0.2 nM T98278 C07CUQ 44311735 IC50 = 0.8 nM T98278 CBW43X 44311736 IC50 = 0.3 nM T98278 CPX02A 44311738 IC50 = 5 nM T98278 CJ2N1I 44311739 IC50 = 3 nM T98278 CA1Y6I 44311752 IC50 = 0.3 nM T98278 CAB87G 44311753 IC50 = 0.2 nM T98278 C8VU6N 44311754 IC50 = 1 nM T98278 C8UXN7 44311755 IC50 = 3 nM T98278 CFZE67 44311758 IC50 = 2 nM T98278 C29QVB 44311775 IC50 = 3 nM T98278 CKF7H2 44311776 IC50 = 3 nM T98278 CT6WL4 44312565 IC50 = 0.47 nM T98278 CQWN95 44312700 IC50 = 44 nM T98278 CLV28B 44314761 IC50 = 0.84 nM T98278 CUIL91 44314780 IC50 = 7.2 nM T98278 CD28FL 44314822 IC50 = 1.2 nM T98278 CJS04N 44314823 IC50 = 0.89 nM T98278 CXDG91 44315057 IC50 = 26.5 nM T98278 C6XVW9 44315058 IC50 = 15 nM T98278 C08CHF 44315059 IC50 = 85 nM T98278 C4VD7T 44315060 IC50 = 33 nM T98278 C2JM6E 44315078 IC50 = 1.9 nM T98278 CF89XK 44315144 IC50 = 1.5 nM T98278 C8S9UP 44315180 IC50 = 12 nM T98278 CH0ZF3 44315282 IC50 = 5.8 nM T98278 C1STV6 44315304 IC50 = 14.7 nM T98278 CTD3M0 44315344 IC50 = 65 nM T98278 CJ4SK0 44315349 IC50 = 18 nM T98278 C8QAE0 44315350 IC50 = 59 nM T98278 CH9Q0J 44315351 IC50 = 1.6 nM T98278 C6BRL3 44316861 IC50 = 298 nM T98278 C9G4AK 44316916 IC50 = 2.9 nM T98278 CWOM31 44317214 IC50 = 48.3 nM T98278 CUY7K1 44325313 Ki = 2.9 nM T98278 C0OYS5 44341922 IC50 = 6 nM T98278 CU14EM 44341923 IC50 = 270 nM T98278 CIQ3Y5 44341924 IC50 = 60 nM T98278 C6AQK3 44341946 IC50 = 24 nM T98278 CK3L7P 44342142 IC50 = 200 nM T98278 C3W0UX 44348523 IC50 = 1 nM T98278 CSO26P 44372686 IC50 = 4 nM T98278 CTRJ86 44372814 IC50 = 15 nM T98278 CQ46VS 44373238 IC50 = 8600 nM T98278 CI8HL6 44404967 IC50 = 13 nM T98278 C4DL5C 44469677 IC50 > 10000 nM T98278 CF31QH 44475015 Ki = 15.85 nM T98278 CB31ST 44726831 IC50 > 79000 nM T98278 C65RAJ 45102601 Ki = 1.259 nM T98278 CG3B8F 45102750 Ki = 0.69 nM T98278 CY05QP 45140560 Ki = 0.7 nM T98278 CG6H2E 45140755 Ki = 31.6 nM T98278 CL2B7W 45140756 Ki = 12.8 nM T98278 CIE1Z6 45141357 Ki = 0.5 nM T98278 CV9GP5 45141358 Ki = 58.2 nM T98278 C0C3AG 45141588 Ki = 3.8 nM T98278 C89QTJ 46184983 IC50 = 12.7 nM T98278 C2R8WH 46232959 IC50 = 288 nM T98278 C3Q6DN 46233002 IC50 > 10000 nM T98278 CH41CI 46835118 IC50 > 79000 nM T98278 C5LJ0V 46835120 IC50 > 79000 nM T98278 CSBO37 46835124 IC50 > 79000 nM T98278 C02ICV 46880542 Ki >= 250 nM T98278 CU2SF8 46880543 Ki >= 250 nM T98278 C6EFX7 46905014 IC50 > 79000 nM T98278 CCUA93 46905018 IC50 > 79000 nM T98278 C85DJM 46905020 IC50 > 79000 nM T98278 CBNT43 46905022 IC50 > 79000 nM T98278 CH20YA 46905025 IC50 > 79000 nM T98278 CWER26 46905028 IC50 > 79000 nM T98278 CD3CK1 46905029 IC50 > 79000 nM T98278 CU6D2Q 46905034 IC50 > 79000 nM T98278 CWY35N 46905037 IC50 > 79000 nM T98278 CP3M2F 46905038 IC50 > 79000 nM T98278 CD47WG 46910493 IC50 = 3.7 nM T98278 C3Y5WG 46910494 IC50 = 22.5 nM T98278 C6ZUA1 46910495 IC50 = 2.6 nM T98278 C4EOT6 46910581 IC50 = 78 nM T98278 CBAG18 46910582 IC50 = 57.6 nM T98278 CF7ID9 46910583 IC50 = 214 nM T98278 C83NXB 46935596 Ki > 10000 nM T98278 CQK7D4 49787115 IC50 > 79000 nM T98278 C86OIB 49787117 IC50 > 79000 nM T98278 CL3D2B 49787119 IC50 > 79000 nM T98278 CP5M7Y 49787120 IC50 > 79000 nM T98278 CW9G1R 49842899 IC50 > 79000 nM T98278 CVC2N3 49842902 IC50 > 79000 nM T98278 C9T3AM 49842903 IC50 > 79000 nM T98278 CQ6V4E 49842905 IC50 > 79000 nM T98278 C62CDL 49842908 IC50 > 79000 nM T98278 C6F2KY 53309128 IC50 = 10.5 nM T98278 C9SA4X 53309129 IC50 = 13.3 nM T98278 C07WMK 53309130 IC50 = 10.2 nM T98278 CLV60X 53309271 IC50 = 8.2 nM T98278 C0SL6H 53309272 IC50 = 202 nM T98278 CBPQ05 53309273 IC50 = 15.7 nM T98278 CR3N6U 53309274 IC50 = 6.8 nM T98278 CA97CK 53309275 IC50 = 16.9 nM T98278 CI6KE2 53309404 IC50 = 3.5 nM T98278 C1EM8J 53309405 IC50 = 748 nM T98278 C0EH4S 53309406 IC50 = 5.2 nM T98278 CG6Z4R 53317942 IC50 = 22 nM T98278 C3U5VH 53319274 Ki = 10 nM T98278 C16BWL 53837978 IC50 = 1100 nM T98278 C0EM7R 54178446 IC50 = 7.6 nM T98278 CG2Z0P 54578725 IC50 = 2.6 nM T98278 CQ3K9X 54693559 IC50 = 0.17 nM T98278 CE75ZL 54768659 IC50 = 2000 nM T98278 CB6FV2 54768660 IC50 = 1600 nM T98278 CBY5V7 54768661 IC50 = 1900 nM T98278 C8ZC6M 54768876 IC50 = 3900 nM T98278 CV4L6Q 54768877 IC50 = 5800 nM T98278 CE8LU3 54771778 IC50 = 2300 nM T98278 C9DMZ4 56964910 Ki > 10000 nM T98278 CW9IF2 57380213 IC50 = 52.5 nM T98278 C20CLX 57380412 IC50 = 2.4 nM T98278 CG09ZX 57380413 IC50 = 326 nM T98278 C19NLI 57380414 IC50 = 4.3 nM T98278 CQ5IJ3 57380415 IC50 = 30.6 nM T98278 C2AVN8 57380416 IC50 = 30.8 nM T98278 CZRA28 57380647 IC50 = 1.3 nM T98278 C5Y1TQ 57380648 IC50 = 106 nM T98278 C52XFK 57380649 IC50 = 198 nM T98278 C1L5WH 60148656 IC50 = 0.7 nM T98278 C5RH7K 60165459 IC50 = 6 nM T98278 CX60UI 67472601 Ki > 10000 nM T98278 C8HRB4 70682146 IC50 = 0.9 nM T98278 CGE5V6 70682147 IC50 = 209 nM T98278 CO58GY 70684248 IC50 = 410 nM T98278 C69ZRA 70684421 IC50 = 630.96 nM T98278 C1PNK9 70686409 IC50 = 19.7 nM T98278 C3GC6L 70686410 IC50 = 1.3 nM T98278 CLH90A 70688502 IC50 = 118.5 nM T98278 CPYZ87 70688503 IC50 = 96.8 nM T98278 C1Q2KU 70688504 IC50 = 37.6 nM T98278 C65DSI 70688681 IC50 = 245 nM T98278 CWP1K8 70690562 IC50 = 78.3 nM T98278 CXK5O2 70690743 IC50 = 117.49 nM T98278 C47THE 70694919 IC50 = 23.99 nM T98278 CCQK74 71456693 IC50 > 79000 nM T98278 CGM32X 71462076 IC50 > 79000 nM T98278 CU73LD 71465043 Ki = 10 nM T98278 CA95RY 71520500 IC50 = 6.8 nM T98278 CGTO05 71520501 IC50 = 7 nM T98278 CQ80JF 71521194 IC50 = 593 nM T98278 CC3F8V 71521195 IC50 = 24.4 nM T98278 CP4W1D 71521196 IC50 = 19.8 nM T98278 CHN49X 71521298 IC50 = 348 nM T98278 C94MCT 71521299 IC50 = 19.4 nM T98278 C9C2NZ 71521300 IC50 = 41 nM T98278 CM79CL 71521301 IC50 = 37.7 nM T98278 CO01SV 71521302 IC50 = 5.1 nM T98278 C5V9UO 71521416 IC50 = 13.5 nM T98278 C89DQL 71521417 IC50 = 94.1 nM T98278 CAT53R 71521418 IC50 = 29.3 nM T98278 CJU56D 71521419 IC50 = 67.4 nM T98278 CM96IV 71521503 IC50 = 36.9 nM T98278 CFA2P7 71521504 IC50 = 81.6 nM T98278 CGN94D 71521505 IC50 = 63.8 nM T98278 CA0K3Z 71521506 IC50 = 45.2 nM T98278 CW1G9U 71521507 IC50 = 250 nM T98278 CPC40O 71521585 IC50 = 63.4 nM T98278 CY4R3B 71623945 IC50 = 293.1 nM T98278 C46YXS 71652853 IC50 = 0.3467 nM T98278 C08SFE 71652855 IC50 = 331.13 nM T98278 CR9B4X 71652857 IC50 = 4.266 nM T98278 CXW1A5 71653008 IC50 = 501.19 nM T98278 CBN4R6 71653151 IC50 = 1698.24 nM T98278 CD79SI 71653304 IC50 = 0.912 nM T98278 C62BDU 71653456 IC50 = 2.884 nM T98278 C8VJ6U 71653747 IC50 = 831.76 nM T98278 CNZ74D 71653749 IC50 = 707.95 nM T98278 CKI9F2 71654379 IC50 = 6456.54 nM T98278 CS0XF8 71654381 IC50 = 42.66 nM T98278 C3HRL4 71717081 IC50 = 416.87 nM T98278 CWH6T3 72548703 IC50 = 0.47 nM T98278 C6EG3T 72697299 Ki > 10000 nM T98278 CIQ29F 72697441 Ki > 10000 nM T98278 CN2GV9 72697443 Ki = 1584.89 nM T98278 CS3I2T 73346386 IC50 = 3 nM T98278 CP2ZR0 73346387 IC50 = 1008 nM T98278 C5L6PQ 73347892 IC50 = 0.4 nM T98278 C4COR6 73347893 IC50 = 0.1 nM T98278 CXYJ62 73349423 IC50 = 1430 nM T98278 CEOK17 73349424 IC50 = 20 nM T98278 CJ6VY2 73350990 IC50 = 115 nM T98278 C2LTU4 73350991 IC50 = 4.9 nM T98278 C7KAB4 73352461 IC50 = 1345 nM T98278 CT1XL6 73352589 Ki > 10000 nM T98278 C9ZC5N 73353933 IC50 = 10 nM T98278 CG71DK 73353934 IC50 = 0.3 nM T98278 CRGQ95 73355474 IC50 = 11 nM T98278 CCEA97 73355475 IC50 = 1.2 nM T98278 CB9DV4 73357016 IC50 = 3.9 nM T98278 CU53JN 73357017 IC50 = 13 nM T98278 C6HJS2 73357018 IC50 = 39 nM T98278 CT9AW2 75031588 Ki = 39.81 nM T98278 C35STH 76310606 IC50 = 128 nM T98278 C18EZQ 76310607 IC50 > 10000 nM T98278 C7DE3L 76310608 IC50 > 10000 nM T98278 CIR72S 76310609 IC50 = 1000 nM T98278 C7IOX1 76310610 IC50 = 60 nM T98278 C2VG1F 76315849 IC50 = 25.4 nM T98278 C9QN4E 76317814 IC50 > 10000 nM T98278 CP7E1N 76317815 IC50 = 97 nM T98278 CS1C9M 76319527 IC50 = 6.1 nM T98278 CD36HB 76321525 IC50 = 23 nM T98278 CZ2I6V 76324571 IC50 = 2.5 nM T98278 CR12QV 76325125 IC50 > 10000 nM T98278 CH1W8N 76325126 IC50 = 1690 nM T98278 C2GY6R 76328690 IC50 = 85 nM T98278 CFNP75 76330043 IC50 = 3.3 nM T98278 C2Q9LU 76330395 IC50 = 9.6 nM T98278 CP4CK9 76333686 IC50 = 29.6 nM T98278 CM4D5H 76333687 IC50 = 2.5 nM T98278 C06XHV 86727577 EC50 = 5100 nM T98278 CK4O2F 87218352 Ki = 50.12 nM T98278 C8O1QX 87218371 Ki = 398.11 nM T98278 C92GXJ 87218373 Ki = 1.259 nM T98278 C8I9AL 87218397 Ki = 630.96 nM T98278 CUT8K1 87218444 Ki = 100 nM T98278 C4BQD9 87218492 Ki = 5.012 nM T98278 C8NEO1 87218514 Ki = 1.259 nM T98278 CR45XW 87218658 Ki = 6.31 nM T98278 C3OGP8 87218678 Ki = 39.81 nM T98278 C0DUB7 87218698 Ki = 5.012 nM T98278 C89OAU 87218826 Ki = 251.19 nM T98278 C1UMO7 87218835 Ki = 31.62 nM T98278 CLIT52 87218933 Ki = 125.89 nM T98278 C2L9SX 87218987 Ki = 19.95 nM T98278 CE09GY 87219028 Ki = 6.31 nM T98278 CREO05 87219032 Ki = 0.7943 nM T98278 C4FML3 87219128 Ki = 125.89 nM T98278 CM96JH 87219174 Ki = 2.512 nM T98278 CM58JI 90219582 EC50 = 5500 nM T98278 C2OQC3 118719137 Ki = 2230 nM T98278 CB0QI8 127026027 IC50 = 87.8 nM T98278 CU0J4F 127026040 IC50 = 69.4 nM T98278 C9QA0N 127026041 IC50 = 67.5 nM T98278 C63KTY 127026042 IC50 = 53.5 nM T98278 C8X0UC 127026043 IC50 = 44 nM T98278 CXN21Q 127026058 IC50 = 347 nM T98278 C4PWU0 127026336 IC50 = 30.7 nM T98278 CFY04E 127026337 IC50 = 93 nM T98278 C5YIM7 127026338 IC50 = 90 nM T98278 C04OWP 127028595 IC50 = 140 nM T98278 CSO5F2 127028617 IC50 = 363 nM T98278 C1OFQ0 127028618 IC50 = 161 nM T98278 C9OW0V 127028619 IC50 = 439 nM T98278 CKY51I 127028620 IC50 = 390 nM T98278 CVKG08 127028930 IC50 = 73.7 nM T98278 CHP7W8 127029201 IC50 = 32.9 nM T98278 CWSI52 127029202 IC50 = 3.9 nM T98278 CH5B3Y 127029203 IC50 = 26.1 nM T98278 CS10YM 127029204 IC50 = 36.9 nM T98278 C36HRE 127030653 EC50 = 1.4 nM T98278 CY0CD4 127030942 Ki = 0.71 nM T98278 C9DO8P 127031265 EC50 = 2.042 nM T98278 CXAG39 127031544 EC50 = 2.344 nM T98278 CHU1J9 127031847 Ki = 9 nM T98278 CEJQ23 127034739 IC50 = 342.8 nM T98278 CU8XB9 127034740 IC50 = 366.3 nM T98278 C5UE4D 127034756 IC50 = 160 nM T98278 CWH4T7 127034757 IC50 = 152 nM T98278 C5E4BU 127034758 IC50 = 13 nM T98278 CGK8W6 127034873 IC50 = 1.1 nM T98278 C7B0JQ 127034874 IC50 = 104 nM T98278 CV4KS1 127034875 IC50 = 93.9 nM T98278 CVK0D7 127034876 IC50 = 106.5 nM T98278 CGVR16 127034901 IC50 = 31 nM T98278 CA15SF 127034903 IC50 = 161.1 nM T98278 CQI70D 127034904 IC50 = 738.4 nM T98278 CF9S8X 127034905 IC50 = 1117.3 nM T98278 CT31NI 127034916 IC50 = 94 nM T98278 CPL08Z 127034917 IC50 = 95 nM T98278 CU39OI 127034918 IC50 = 373 nM T98278 C64HFO 127034919 IC50 = 341 nM T98278 CN7DB6 127034920 IC50 = 57.4 nM T98278 CQOV56 127034921 IC50 = 7.3 nM T98278 CRF7J1 127034922 IC50 = 6.3 nM T98278 CZ61LK 127034966 EC50 > 5011.87 nM T98278 CA0SN5 127034967 EC50 > 5011.87 nM T98278 C5XM0K 127035067 IC50 = 47 nM T98278 C1QJ0V 127035068 IC50 = 201 nM T98278 CBC74Y 127035069 IC50 = 419 nM T98278 C67FNJ 127035070 IC50 = 28 nM T98278 CL01XK 127035082 IC50 = 50 nM T98278 CP6T3J 127035083 IC50 = 81 nM T98278 CJHG08 127035084 IC50 = 56 nM T98278 CLJ94G 127035085 IC50 = 8 nM T98278 CRN65G 127035219 IC50 = 217 nM T98278 C83ZIH 127035246 IC50 = 3.5 nM T98278 CQV63D 127035247 IC50 = 1368.1 nM T98278 C6JTW5 127035248 IC50 = 609.2 nM T98278 C9RCI8 127035249 IC50 = 699.3 nM T98278 C3AJ4Z 127035263 IC50 = 61.2 nM T98278 C7OE8P 127035264 IC50 = 2.7 nM T98278 C6CP8U 127035265 IC50 = 1.4 nM T98278 CE07IC 127035379 IC50 = 42 nM T98278 C6DU4R 127035380 IC50 = 76 nM T98278 C9S4JW 127035381 IC50 = 671.4 nM T98278 C75KYB 127035391 IC50 = 788.4 nM T98278 C2NX4L 127035392 IC50 = 486.8 nM T98278 CP30HO 127035393 IC50 = 621.6 nM T98278 C3XWN4 127035410 IC50 = 16 nM T98278 CHN1I9 127035514 IC50 = 156.8 nM T98278 CIKB36 127035515 IC50 = 38.9 nM T98278 CA9FD3 127035544 IC50 = 37 nM T98278 CF6X3E 127035545 IC50 = 92 nM T98278 CHWP78 127035557 IC50 = 503.3 nM T98278 C2SI6O 127035558 IC50 = 87.2 nM T98278 CRAX67 127035715 IC50 = 40.4 nM T98278 C1BZJ5 127035716 IC50 = 23 nM T98278 CZM6R9 127035717 IC50 = 5 nM T98278 C5ED6S 127035757 IC50 = 7 nM T98278 CD0T4M 127036102 IC50 = 19.5 nM T98278 CW6Z5T 127036103 IC50 = 90.5 nM T98278 C5E6QH 127036104 IC50 = 1534.5 nM T98278 C2E0ZQ 127036105 IC50 = 495.8 nM T98278 C3WQD1 127036106 IC50 = 128.6 nM T98278 CNX0J3 127036107 IC50 = 57.9 nM T98278 CR1YG9 127036108 IC50 = 70 nM T98278 CQLC17 127036294 IC50 = 1536.6 nM T98278 C63ZGR 127036297 IC50 = 214.4 nM T98278 CZN92T 127036865 IC50 = 82 nM T98278 C0KJO7 127036866 IC50 = 73.3 nM T98278 C19VDE 127036867 IC50 = 53.9 nM T98278 C24HFS 127036868 IC50 = 549.8 nM T98278 CPQB01 127037496 IC50 = 465 nM T98278 CEQS03 127037497 IC50 = 385 nM T98278 CW8QT1 137527725 IC50 >= 10 nM T98278 C2ND9V 137532858 IC50 = 1.6 nM T98278 C7KD9N 142533975 IC50 = 2.2 nM T98278 C6Z9HB 142534004 IC50 = 38 nM T98278 C8UL6O 142534045 IC50 = 0.7 nM T98278 C9UR5L 142534050 IC50 = 2 nM T98278 CKV4L6 142534121 IC50 = 2.1 nM T98278 C5ZXV2 142534141 IC50 = 1.2 nM T98278 C9AS2D 142534170 IC50 = 32 nM T98278 CXJ8M1 142534183 IC50 = 4.7 nM T98278 C9HAT3 142534191 IC50 = 5.6 nM T98278 CGM6C1 145925549 EC50 = 44 nM T98278 CF8I6Q 145948674 Ki = 13 nM T98278 CQBU72 145952582 Ki = 317 nM T98278 CI2M1Q 145957579 Ki = 24838 nM T98278 CKGV06 145957897 Ki = 1.35 nM T98278 C8QL0G 145981239 IC50 = 1.8 nM T98278 CQB9O0 145987183 IC50 = 70 nM T98278 CG6KB7 155512629 Ki = 7.943 nM T98278 C9KP4F 155513439 Ki = 79.43 nM T98278 C1HOG5 155514738 Ki = 10 nM T98278 CN7Z5E 155516694 Ki = 199.53 nM T98278 C1PUC8 155517399 IC50 = 2.2 nM T98278 C21TUL 155520317 Ki = 125.89 nM T98278 CX1YU9 155522135 Ki = 398.11 nM T98278 C30EFX 155523092 Ki = 125.89 nM T98278 C7WI9L 155526996 Ki = 31.62 nM T98278 C1G7LY 155529942 Ki = 50.12 nM T98278 CVXJ96 155533580 Ki = 63.1 nM T98278 CNV2A8 155535176 Ki = 158.49 nM T98278 C5D3AP 155542482 IC50 = 1.5 nM T98278 CFM26N 155547799 Ki = 50.12 nM T98278 C5AF2L 155551279 EC50 = 17 nM T98278 C1RUT3 155552503 Ki = 31.62 nM T98278 CUE8Y9 155557693 Ki = 15.85 nM T98278 CS7ZV8 155565351 Ki = 79.43 nM T98278 D00LWG 46880545 Ki = 0.7 nM T98278 D04SVT 9829012 IC50 = 0.1 nM T98278 D05NXX 7217941 IC50 > 79000 nM T98278 D06DRC 45141142 Ki = 0.3 nM T98278 D06PJZ 45140373 Ki = 0.6 nM T98278 D07EWK 46880541 Ki = 0.4 nM T98278 D0A4NO 6603900 IC50 = 1.1 nM T98278 D0D1FT 108185 IC50 = 2 nM T98278 D0K2EX 9804984 Ki = 10000 nM T98278 D0L3PY 123814 Ki = 407.38 nM T98278 D0M5ZE 5311416 Ki < 10000 nM T98278 D0MH1K 9935096 IC50 = 4.9 nM T98278 D0N2WA 46880540 Ki = 0.8 nM T98278 D0O0SH 9932483 IC50 = 6.5 nM T98278 D0O1YO 45140942 Ki = 0.4 nM T98278 D0PB5Q 3132 Ki > 10000 nM T98278 D0U7QE 45140941 Ki = 0.7 nM T98278 D0XO1T 46880544 Ki = 0.6 nM T98278 D0Z7AF 10031067 IC50 = 2.1 nM T67619 D00FGR 3599 IC50 = 9600 nM T67619 D03MNN 11341869 IC50 > 1000 nM T67619 D0EG1I 9926791 IC50 > 10000 nM T67619 D0J9ZR 4477 IC50 = 59400 nM T67619 D0K8KX 5280343 IC50 = 5390 nM T67619 D0R0MW 5329102 IC50 > 10000 nM T67619 D01NEC 51042438 IC50 = 18 nM T67619 D01ZAQ 25227436 IC50 = 3 nM T67619 D02RJY 11442891 IC50 > 10000 nM T67619 D02ZQS 16095342 IC50 = 955 nM T67619 D03BBG 46843057 Ki = 0.08 nM T67619 D03HUX 49792852 IC50 > 10000 nM T67619 D03LWG 53235510 IC50 > 10000 nM T67619 D07EHV 44814409 IC50 > 10000 nM T67619 D07HPJ 11476171 IC50 > 10000 nM T67619 D08QGT 17755052 IC50 = 37 nM T67619 D09IYM 24905401 IC50 = 38 nM T67619 D09XZL 56962369 IC50 < 1 nM T67619 D0CY1B 6420138 Ki > 10000 nM T67619 D0E3TC 44259 IC50 = 1.5 nM T67619 D0I4TH 24788740 IC50 = 157 nM T67619 D0L4FS 5280961 IC50 > 70000 nM T67619 D0M9QZ 11485656 IC50 = 50000 nM T67619 D0MS3Z 16725726 Ki = 1 nM T67619 D0N5JZ 25033539 IC50 = 13 nM T67619 D0O0LS 25141092 IC50 > 10000 nM T67619 D0P1CV 46191454 IC50 > 10000 nM T67619 D0Q9UX 16718576 IC50 > 10000 nM T67619 D0R1VU 148177 IC50 = 5300 nM T67619 D0W3RW 24964624 IC50 = 8 nM T67619 D0X2JM 56963011 IC50 = 1 nM T67619 D0Z1DH 10029385 IC50 > 20000 nM T67619 D03BNU 59604787 IC50 > 3500 nM T67619 D0LF0O 135441202 IC50 = 48390 nM T67619 D0YK9D 9956119 IC50 > 10000 nM T67619 D0ZE5U 11161844 IC50 = 100 nM T67619 D0T3ME 156422 IC50 > 30000 nM T67619 CX02HJ 1392 IC50 = 3500 nM T67619 C2BR0H 9221 IC50 > 398107.17 nM T67619 COYW98 9222 IC50 > 400000 nM T67619 C3FD6V 13028 IC50 = 12270 nM T67619 C5CYL1 25450 IC50 = 313 nM T67619 C63WLY 89644 IC50 = 6.7 ug.mL-1 T67619 C5JE2Z 104860 IC50 > 10 ug.mL-1 T67619 C3XD4Z 139106 IC50 = 135000 nM T67619 C5EH9L 139601 IC50 = 80000 nM T67619 CI1NA5 159926 IC50 > 10 ug.mL-1 T67619 C2L9OS 163292 IC50 = 198 nM T67619 CYBA43 177458 IC50 > 10 ug.mL-1 T67619 C29FQA 234762 IC50 = 20000 nM T67619 CHEZ24 399491 IC50 = 54480 nM T67619 CN05AH 406563 IC50 > 10000 nM T67619 C4MNG8 445840 IC50 > 10000 nM T67619 C1ZG2U 449087 IC50 > 10000 nM T67619 CJ75ZW 657581 IC50 = 20000 nM T67619 CJ7KT3 694845 IC50 > 50000 nM T67619 C6IW2P 1131425 IC50 = 60200 nM T67619 C0BZG7 1207540 IC50 = 126000 nM T67619 C10TNL 1270181 Ki = 20800 nM T67619 C8KPM0 1776570 Ki = 1100 nM T67619 C1SVD2 2132479 IC50 = 2600 nM T67619 C86LNP 2779952 IC50 > 100000 nM T67619 C1J3AU 2810537 IC50 > 50000 nM T67619 CTR7H2 3084051 IC50 = 424 nM T67619 CCOU85 3800302 IC50 = 25000 nM T67619 CEU1N6 5056270 IC50 > 20000 nM T67619 C8IAR2 5281657 IC50 > 100000 nM T67619 CI68PW 5283685 IC50 > 100000 nM T67619 CXK0S6 5283727 IC50 > 100000 nM T67619 C31FHN 5330788 IC50 = 5480 nM T67619 CS94ZR 5343381 Ki = 3900 nM T67619 CDQ3M7 5359485 IC50 > 10 ug.mL-1 T67619 C54BYP 5360741 IC50 = 7.9 ug.mL-1 T67619 CDK3J0 5703619 IC50 = 11 nM T67619 CYTV91 6443339 IC50 = 143900 nM T67619 CG17TN 6914611 Ki = 2 nM T67619 C7E2QK 6914613 IC50 = 14 nM T67619 CW9X0N 6914614 IC50 = 190 nM T67619 C4G9WR 9547398 IC50 > 100000 nM T67619 C76CUP 9547698 IC50 > 100000 nM T67619 CQ57EC 9548013 IC50 > 100000 nM T67619 CIAL53 9819282 IC50 = 3400 nM T67619 CC7Y2O 9828163 IC50 = 45 nM T67619 C8QZD6 9829528 IC50 = 3.8 nM T67619 CM5Z8X 9869943 IC50 > 1000 nM T67619 CI0AW6 9871034 IC50 = 290 nM T67619 C7H8EO 9871171 IC50 = 86 nM T67619 C18HKQ 9885748 IC50 = 780 nM T67619 CUE4B5 9912061 IC50 = 1288 nM T67619 C5GE7T 9917045 IC50 = 6400 nM T67619 CJO47T 9948405 IC50 > 10000 nM T67619 CU7FH2 9957031 IC50 = 762 nM T67619 CV8I5X 9999342 IC50 > 10000 nM T67619 CR8DA1 10024683 IC50 > 100000 nM T67619 CLA93G 10047202 IC50 > 100000 nM T67619 C3LCH5 10047545 IC50 > 100000 nM T67619 C7YD1X 10048045 IC50 > 25000 nM T67619 CJX43Z 10055074 IC50 = 458 nM T67619 CJT0V2 10062782 IC50 = 5290 nM T67619 C0AH5W 10126464 IC50 = 1.5 nM T67619 CYX37N 10126724 IC50 = 227 nM T67619 CF30QE 10127189 IC50 = 12 nM T67619 C7GJ3H 10127292 IC50 = 32250 nM T67619 CBY3F2 10127782 IC50 = 9.8 nM T67619 CEV18B 10128689 IC50 = 17000 nM T67619 CTA2P0 10150362 IC50 = 360 nM T67619 CBW7U5 10150682 IC50 = 300 nM T67619 CVSX67 10150925 IC50 = 1.15 nM T67619 C7PK4U 10152003 IC50 = 3029 nM T67619 C4FUG5 10152760 IC50 > 50000 nM T67619 CMO32F 10152761 IC50 = 21200 nM T67619 CB1K2O 10172517 IC50 = 9.7 nM T67619 C7R5DM 10172543 IC50 = 24010 nM T67619 CPQT23 10172738 IC50 = 278 nM T67619 CD1O8L 10172789 IC50 = 1659 nM T67619 C9IM0S 10172981 IC50 = 12030 nM T67619 CS9J2F 10173098 IC50 = 270 nM T67619 CU0GF4 10173112 IC50 = 210 nM T67619 C3N4PB 10173974 IC50 = 1.3 nM T67619 CMR17F 10174144 IC50 = 1500 nM T67619 CN01JZ 10193747 IC50 = 1560 nM T67619 CJLT23 10194089 IC50 = 31280 nM T67619 CQRS02 10194205 IC50 = 26 nM T67619 CTC89D 10194362 IC50 = 23 nM T67619 CLP79V 10196532 IC50 = 166 nM T67619 CU15MK 10215707 IC50 = 1830 nM T67619 CQ1E6B 10216067 IC50 = 331 nM T67619 CGT7V4 10216158 IC50 = 179 nM T67619 CI8MW4 10216627 IC50 = 1.8 nM T67619 C52HOJ 10216834 IC50 = 6230 nM T67619 C7X2SF 10217131 IC50 = 3.9 nM T67619 C0O8FI 10217663 IC50 = 1003 nM T67619 CY6MJ3 10218178 IC50 > 50000 nM T67619 CT97JL 10218280 IC50 = 244 nM T67619 C36MZO 10237197 IC50 = 210 nM T67619 C21-DEC 10237270 IC50 = 4022 nM T67619 CZ39AX 10237559 IC50 = 1117 nM T67619 CH1A8K 10237631 IC50 = 3.2 nM T67619 C3V5CX 10237634 IC50 = 2.9 nM T67619 C92GEF 10237709 IC50 = 198 nM T67619 C70OSH 10237750 IC50 = 273 nM T67619 C42QYD 10238049 IC50 = 2.6 nM T67619 C96QHV 10238471 IC50 = 2710 nM T67619 C9K1CJ 10238690 IC50 = 18 nM T67619 C8V6RI 10240275 IC50 = 253 nM T67619 C5TQ7X 10247543 IC50 > 10000 nM T67619 CDKN83 10247683 Ki = 1525 nM T67619 C6LHG1 10287346 IC50 = 142 nM T67619 C50LNE 10287431 IC50 = 7090 nM T67619 CS4AV1 10287447 IC50 = 215 nM T67619 C6FX3E 10287639 IC50 = 273 nM T67619 CZ5UN3 10287988 IC50 = 407 nM T67619 CU12EK 10288118 IC50 = 3670 nM T67619 CD3W6Y 10289038 Ki = 760 nM T67619 C65DNI 10289089 IC50 = 1450 nM T67619 C2LP9A 10289671 IC50 = 85 nM T67619 C7SFI1 10296883 IC50 > 10000 nM T67619 CJ7RM2 10309064 IC50 = 6940 nM T67619 C36MFC 10309109 IC50 = 4040 nM T67619 CEV5Z1 10309398 IC50 = 146 nM T67619 C5QE3H 10309844 IC50 = 1022 nM T67619 CU18ZF 10310117 IC50 = 18 nM T67619 CT0M7Q 10311653 IC50 = 1834 nM T67619 C4MOF8 10312133 IC50 = 20 nM T67619 CAK9U4 10415819 IC50 = 63 nM T67619 C4CP7K 10423452 IC50 > 100000 nM T67619 C40AJH 10428289 Ki = 89.6 nM T67619 C7HBP6 10429593 IC50 > 10000 nM T67619 C2WQ8M 10473563 IC50 > 10000 nM T67619 C1XL3P 10475646 IC50 = 29 nM T67619 CEML49 10538870 IC50 > 100000 nM T67619 C9O2PG 10588346 IC50 > 100000 nM T67619 C7KF2E 10705154 IC50 = 92000 nM T67619 C83QWV 10714343 IC50 = 48400 nM T67619 C2C8GH 10732141 IC50 > 100000 nM T67619 C5R7EZ 10901296 IC50 = 2940 nM T67619 C53MZX 11168481 IC50 = 763 nM T67619 C3IJ6D 11180030 IC50 = 6915 nM T67619 CPVK21 11180486 IC50 = 131 nM T67619 C8G5WP 11210533 IC50 = 4070 nM T67619 C7BN5E 11225451 IC50 = 2874 nM T67619 CC6V3Z 11225497 IC50 = 46 nM T67619 C1UZC6 11226082 IC50 = 5548 nM T67619 C8Y6IM 11234514 IC50 = 94 nM T67619 CKB72H 11237628 IC50 = 2249 nM T67619 CRG03D 11245934 IC50 = 331 nM T67619 C2ON6C 11246455 IC50 = 20 nM T67619 C30PKR 11248978 IC50 > 20000 nM T67619 CCF0G6 11249067 IC50 = 495 nM T67619 C49NET 11256399 IC50 = 56 nM T67619 C1TCF3 11260243 IC50 = 7407 nM T67619 COHW29 11272514 IC50 = 273 nM T67619 CBOP58 11293798 Ki = 1070 nM T67619 CSXY78 11294864 IC50 > 20000 nM T67619 CHBC32 11296432 IC50 = 21 nM T67619 CPU9I3 11316975 IC50 > 20000 nM T67619 C7E5OS 11327794 IC50 = 0.6 nM T67619 CQ8I4H 11328863 IC50 > 20000 nM T67619 CPV82H 11341558 IC50 = 239 nM T67619 C8XIF5 11350077 IC50 = 77 nM T67619 CRTG16 11359538 IC50 = 15000 nM T67619 C26BZX 11362471 Ki = 3150 nM T67619 C4G3RZ 11364261 IC50 = 4237 nM T67619 C1LT9H 11374804 IC50 = 4397 nM T67619 CWXB93 11397177 Ki > 10000 nM T67619 CPFW90 11399527 IC50 = 121 nM T67619 CWM18I 11406175 IC50 = 9210 nM T67619 C6KQ2U 11409661 IC50 = 3323 nM T67619 C4L5TF 11409804 IC50 = 253 nM T67619 C1WXC5 11417488 IC50 > 50000 nM T67619 C0APW4 11422034 IC50 > 10000 nM T67619 C1FC5U 11431759 IC50 = 865 nM T67619 C64IGY 11448608 Ki > 5000 nM T67619 CI9L2T 11454186 IC50 = 1471 nM T67619 CQS3U5 11454871 IC50 = 177 nM T67619 CE72WO 11489421 IC50 = 8457 nM T67619 C17UMV 11495551 IC50 = 10 nM T67619 C7XM4C 11504922 IC50 = 24 nM T67619 C3D9OU 11509538 IC50 = 47 nM T67619 CCX5Y9 11509539 IC50 = 19 nM T67619 CPN02A 11513279 IC50 = 9 nM T67619 C38OKZ 11513374 IC50 = 13 nM T67619 C3VXY4 11518055 IC50 = 79 nM T67619 CU79NQ 11524833 IC50 = 357 nM T67619 CJ7XT8 11526364 IC50 = 81 nM T67619 CTM2Q3 11526695 IC50 = 21 nM T67619 C7HMO6 11526786 IC50 > 30000 nM T67619 CEX8Y5 11527102 IC50 = 7 nM T67619 CL7X4Q 11530963 IC50 > 100000 nM T67619 C5NPU9 11534762 IC50 = 286 nM T67619 CRPL63 11538974 IC50 = 25 nM T67619 CJIW92 11539281 IC50 = 6.1 nM T67619 CTG83F 11539329 Ki > 8200 nM T67619 CG84SZ 11540975 IC50 = 8.5 nM T67619 CWCN15 11541348 IC50 = 4 nM T67619 CY0JX9 11541985 IC50 = 44 nM T67619 CSCJ29 11542208 IC50 = 36 nM T67619 CA8R0K 11547290 IC50 = 560 nM T67619 CX96EC 11549174 IC50 = 10 nM T67619 C3Z8PI 11549180 IC50 = 9 nM T67619 CJEB45 11549190 IC50 = 91 nM T67619 CJF21M 11549537 IC50 = 38 nM T67619 CJ8BQ6 11552741 IC50 = 24 nM T67619 CN25UD 11556452 IC50 = 14 nM T67619 CACS26 11561968 Ki > 10000 nM T67619 C45QDX 11568147 IC50 = 3 nM T67619 C4AL8Z 11575817 IC50 = 79 nM T67619 C9LDN1 11577612 IC50 = 42.6 nM T67619 C0B2EI 11581739 IC50 = 38 nM T67619 C9EIF4 11582467 IC50 = 6 nM T67619 CO9KP5 11583459 IC50 > 10000 nM T67619 CPJZ24 11584546 IC50 = 129 nM T67619 C0SCK2 11585287 IC50 = 765 nM T67619 CMIL86 11590363 Ki > 8200 nM T67619 C6C0VR 11592032 IC50 = 9.7 nM T67619 CK61VI 11606572 IC50 = 96.4 nM T67619 C20IRX 11606613 IC50 = 64 nM T67619 C7PA8T 11607451 IC50 = 6 nM T67619 C5XC9Q 11611566 IC50 = 15 nM T67619 C3FQP1 11614515 IC50 = 4 nM T67619 CBEG76 11621110 IC50 = 4.5 nM T67619 C3NDK9 11633229 IC50 = 790 nM T67619 CP2R3O 11636277 IC50 = 7 nM T67619 C4YWT2 11636404 IC50 = 3 nM T67619 CABL68 11639899 IC50 = 8.9 nM T67619 C9T6SC 11640926 Ki > 8200 nM T67619 C2OC8S 11642946 IC50 = 5 nM T67619 CDY01B 11643074 IC50 = 75 nM T67619 C9RLC8 11643116 IC50 = 46 nM T67619 CP0I2U 11643417 IC50 = 8 nM T67619 C4GTZ8 11645322 IC50 > 20000 nM T67619 CM08LS 11648365 IC50 = 100 nM T67619 CPA5Y7 11650332 IC50 = 42 nM T67619 COR9B8 11650399 IC50 = 5 nM T67619 CCH38R 11654950 IC50 = 18 nM T67619 C87JQN 11663666 IC50 = 69 nM T67619 C7XEV0 11664023 IC50 = 6 nM T67619 CESQ80 11670972 IC50 = 18 nM T67619 C43LDG 11671553 IC50 = 5 nM T67619 CTI6U1 11671757 IC50 = 17 nM T67619 CX1GS0 11672017 IC50 = 3 nM T67619 CON70D 11672049 IC50 = 33 nM T67619 C0V7SU 11675388 IC50 = 13 nM T67619 C9G3OH 11675718 IC50 = 14 nM T67619 COEL03 11676096 IC50 = 40 nM T67619 CU0E8O 11690457 Ki > 10000 nM T67619 C25STN 11690618 IC50 = 50 nM T67619 C81CLV 11693440 IC50 = 19 nM T67619 CA78WD 11702853 IC50 = 4.8 nM T67619 C0NRG1 11703456 IC50 = 0.59 nM T67619 CB0AP2 11705863 Ki > 10000 nM T67619 CCK3Q5 11712132 IC50 = 99 nM T67619 CY8U0T 11713130 IC50 = 15 nM T67619 CY8C9P 11751126 IC50 = 33 nM T67619 CP7AH3 11755812 IC50 = 50000 nM T67619 CHD8K3 11774303 IC50 = 138 nM T67619 C9JT4S 11847343 IC50 > 10000 nM T67619 C9A6KM 11857236 Ki = 0.2 nM T67619 CHR92S 11858109 IC50 > 100000 nM T67619 CA9ST2 11959186 IC50 = 13 nM T67619 CC7M0D 11959190 IC50 = 8 nM T67619 C39VTW 11959283 IC50 = 6 nM T67619 CQ8U1P 11959284 IC50 = 3 nM T67619 C36HDX 11959286 IC50 = 3 nM T67619 CTE96C 11959310 IC50 = 4 nM T67619 CO0A4K 11959314 Ki = 0.4 nM T67619 C12CRJ 11959377 IC50 = 6 nM T67619 CUWL12 11959378 IC50 = 2 nM T67619 CVPT94 11959513 IC50 = 63 nM T67619 C5LZ9C 11959550 IC50 = 16 nM T67619 C3UVQ2 11959600 IC50 = 12 nM T67619 C1WDQ0 11959682 IC50 = 5 nM T67619 CMW89V 11959683 IC50 = 3 nM T67619 CA6K4Y 11959684 IC50 = 3 nM T67619 CZ2L6M 11995746 IC50 = 5.8 nM T67619 C9VHS4 11996315 IC50 = 4.8 nM T67619 CB36UI 11996316 IC50 = 96 nM T67619 C70MRY 11996623 IC50 = 2 nM T67619 CFY6V4 11996779 IC50 = 75 nM T67619 CF4KG0 12118709 IC50 > 100000 nM T67619 C90OYV 14044888 IC50 = 50000 nM T67619 CO1L4P 14332591 IC50 > 100000 nM T67619 C96NWB 14604081 IC50 = 5400 nM T67619 CDGF78 15282555 IC50 = 1900 nM T67619 C3FEG7 15296047 IC50 = 580 nM T67619 C7N6CQ 15604547 IC50 = 930 nM T67619 C5SA9D 15929390 IC50 > 100000 nM T67619 CSA02I 15979148 IC50 = 4.6 nM T67619 CBE54Y 15979149 IC50 = 27 nM T67619 C9YE7I 15979150 IC50 = 18.3 nM T67619 C92FEN 15979151 IC50 = 17 nM T67619 C9QO8U 15979276 IC50 = 4 nM T67619 CFPW41 16007116 Ki > 8200 nM T67619 CLE26B 16037748 Ki = 3282 nM T67619 CAR74L 16040274 IC50 = 0.6 nM T67619 CZK8V6 16043304 IC50 = 6 nM T67619 C9TU1O 16046126 IC50 > 1000 nM T67619 CZHJ34 16058637 IC50 = 15000 nM T67619 C3G6HX 16058667 Ki = 80 nM T67619 C3VA5P 16066787 IC50 = 11800 nM T67619 CKV4G1 16079040 IC50 = 20 nM T67619 CKR57M 16086104 IC50 > 25000 nM T67619 C16NRY 16086114 IC50 > 25000 nM T67619 CBM80K 16091080 IC50 = 2.8 nM T67619 C7Z4LV 16095343 IC50 = 324 nM T67619 CQG45C 16109001 IC50 = 100000 nM T67619 CBA2W5 16122641 IC50 = 1360 nM T67619 CD41WU 16122642 IC50 = 5 nM T67619 C9IW5S 16730105 IC50 > 100000 nM T67619 C0H8UN 16730109 IC50 > 50000 nM T67619 C2H4LM 16731495 IC50 = 20.7 nM T67619 CI7X5O 16731496 IC50 = 10 nM T67619 CFU05S 16731497 IC50 = 1.3 nM T67619 CTP46K 16731498 IC50 = 49 nM T67619 CO07TD 16731499 IC50 = 3.9 nM T67619 CS7A4O 16731500 IC50 = 2.5 nM T67619 C7QDY2 16731501 IC50 = 11 nM T67619 CMV8Q3 16731503 IC50 = 15.3 nM T67619 CR2X8K 16731505 IC50 = 20.3 nM T67619 CJ3VT4 16731507 IC50 = 126 nM T67619 CH68OM 16731509 IC50 = 14 nM T67619 CRU83C 16731662 IC50 = 6 nM T67619 C7MED6 16731663 IC50 = 6.8 nM T67619 C8V4QA 16731664 IC50 = 78 nM T67619 C4A7ZI 16731671 IC50 = 751 nM T67619 CVNA25 16731834 IC50 = 47 nM T67619 CH6MD7 16731836 IC50 = 0.6 nM T67619 COY7P8 16731838 IC50 = 7.2 nM T67619 C87WEG 16731841 IC50 = 5 nM T67619 CID78A 16731843 IC50 = 16 nM T67619 C0OWL3 16731987 IC50 = 1.4 nM T67619 CZM0A2 16731988 IC50 = 8.4 nM T67619 C4EP1U 16731989 IC50 = 21 nM T67619 C21-AUG 16731990 IC50 = 31 nM T67619 CNKF23 16731991 IC50 = 5.9 nM T67619 CL4N9F 16731992 IC50 = 23 nM T67619 CHI7J1 16732132 IC50 = 3.6 nM T67619 C9T4VW 16732276 IC50 = 2.9 nM T67619 CA6CE1 16732278 IC50 = 39 nM T67619 C57GQS 16732279 IC50 = 1.2 nM T67619 CH76CW 16732414 IC50 = 1.8 nM T67619 C5L4AJ 16732415 IC50 = 1.2 nM T67619 CQ2AP4 16732416 IC50 = 12.1 nM T67619 C1C3SJ 16732417 IC50 = 3.3 nM T67619 C1L7KM 16732418 IC50 = 42 nM T67619 CC9N3K 16732419 IC50 = 13 nM T67619 CW72NH 16732420 IC50 = 290 nM T67619 CA2K9Y 16732881 IC50 = 8.5 nM T67619 CZH6E0 16732883 IC50 = 65.5 nM T67619 CFA4T7 16733021 IC50 = 11 nM T67619 CP25BF 16733023 IC50 = 2.1 nM T67619 CPT94S 16733025 IC50 = 0.9 nM T67619 CXUL72 16733027 IC50 = 5.6 nM T67619 CUZE96 16733156 IC50 = 12 nM T67619 CEJ7I4 16733278 IC50 = 2.4 nM T67619 C0XL5Q 16733284 IC50 = 3.1 nM T67619 C7LI4T 16733286 IC50 = 57 nM T67619 C8YT6P 16733397 IC50 = 7.7 nM T67619 CQT6Z7 16733398 IC50 = 18 nM T67619 CT79UJ 16733399 IC50 = 13.3 nM T67619 CF7EV9 16733400 IC50 = 3.1 nM T67619 C8MES6 16733403 IC50 = 1.8 nM T67619 C0O6SY 17751068 IC50 = 1.9 nM T67619 C9C5TV 17751819 IC50 = 0.66 nM T67619 CVS0T5 17754396 IC50 > 10000 nM T67619 C5DK1N 18458970 IC50 = 10870 nM T67619 CIW74O 18963535 IC50 > 50000 nM T67619 CHV89K 20744784 IC50 = 260 nM T67619 C2ZNX3 20744789 IC50 = 121 nM T67619 C80DGN 20744797 IC50 = 500 nM T67619 CBV17Q 20744799 IC50 = 324 nM T67619 C5CE1L 20744801 IC50 = 320 nM T67619 CXDB30 20744806 IC50 = 19320 nM T67619 C32HPS 20744808 IC50 = 690 nM T67619 C7SL1T 20744810 IC50 = 1100 nM T67619 CL81VC 21100709 IC50 = 38600 nM T67619 CWK2H5 21103101 IC50 = 107 nM T67619 CA46OM 21103107 IC50 = 365 nM T67619 CJXU82 21103111 IC50 = 1089 nM T67619 CF9YE6 21103119 IC50 = 55 nM T67619 C5AR9M 21103197 IC50 = 240 nM T67619 C2Y3IB 21147597 IC50 = 3900 nM T67619 CLH26A 22607234 IC50 = 14710 nM T67619 C71FSD 22607483 IC50 = 14710 nM T67619 C2CD7W 22872615 IC50 = 10870 nM T67619 CQ3DK7 22961870 IC50 = 23910 nM T67619 C6RG5Y 23644684 IC50 = 33160 nM T67619 CRW1H5 23644685 Ki = 465 nM T67619 C0W8LS 23645850 IC50 = 4 nM T67619 C6HC1V 23646944 IC50 = 25200 nM T67619 CX19VS 23646949 IC50 = 9870 nM T67619 C3PW2A 23646950 IC50 = 9350 nM T67619 C1FKW6 23646951 IC50 = 2860 nM T67619 CAG31D 23646952 IC50 = 2160 nM T67619 CMX3Q5 23646953 IC50 = 18830 nM T67619 C91VPI 23646954 IC50 = 6970 nM T67619 CA6D1B 23646955 IC50 = 31950 nM T67619 CK4FB0 23646956 IC50 = 1340 nM T67619 CQAW67 23646958 IC50 = 9310 nM T67619 C3O2AT 23646963 IC50 = 1390 nM T67619 CW8X0Q 23646965 IC50 = 33010 nM T67619 C34BSP 23646966 IC50 = 1120 nM T67619 CNU42R 23646967 IC50 = 14330 nM T67619 CQG0R4 23646968 IC50 = 2170 nM T67619 CHP17G 23646970 IC50 = 8020 nM T67619 CB7L9J 23646972 IC50 = 875 nM T67619 CFWC43 23646973 IC50 > 50000 nM T67619 CGJ6S9 23646974 IC50 = 19 nM T67619 CPS34L 23646975 IC50 = 79 nM T67619 CF0QK9 23646977 IC50 = 3200 nM T67619 C4UA8R 23646978 IC50 = 668 nM T67619 CP04EG 23646979 IC50 = 284 nM T67619 C6HW1C 23646980 IC50 = 760 nM T67619 C42WRI 23646984 IC50 = 23270 nM T67619 CAK6T0 23646986 IC50 = 43010 nM T67619 CJ9T1S 23646987 IC50 = 2670 nM T67619 CQ3O5D 23646988 IC50 = 6450 nM T67619 CJR8L7 23646989 IC50 = 6350 nM T67619 C5H9MJ 23646990 IC50 = 3110 nM T67619 C0KPN4 23646991 IC50 = 176 nM T67619 CZQ53I 23646992 IC50 = 163 nM T67619 C5NQ9I 23646993 IC50 = 69 nM T67619 CW2L3O 23646994 IC50 = 147 nM T67619 C4K2BJ 23646995 IC50 = 3340 nM T67619 COF3T4 23646996 Ki = 54.6 nM T67619 C5E3ZD 23646997 Ki = 6.8 nM T67619 C8RIO0 23646998 Ki = 63.7 nM T67619 CX2IO1 23646999 Ki = 3.5 nM T67619 C9JXP5 23647000 Ki = 85 nM T67619 CPS28V 23647001 Ki = 672 nM T67619 CBI65P 23647002 Ki = 2.1 nM T67619 CNET21 23647003 Ki = 6.6 nM T67619 CG6P5Q 23647004 Ki = 3.2 nM T67619 CBDN19 23647005 Ki = 8.3 nM T67619 C31JYB 23647006 Ki = 1.1 nM T67619 CFLN54 23647007 Ki = 185 nM T67619 CW4O2P 23647008 Ki = 368 nM T67619 C8NYV0 23647009 Ki = 233 nM T67619 C5HXS9 23647010 Ki = 289 nM T67619 CKH3B9 23647011 Ki = 197 nM T67619 CV7FX6 23647012 Ki = 70.6 nM T67619 CSVI73 23647013 Ki = 8.3 nM T67619 C04GFC 23647014 Ki = 244 nM T67619 CUYT34 23647015 Ki = 626 nM T67619 CN1O7X 23647016 IC50 = 17000 nM T67619 CJ3EO0 23647017 IC50 > 50000 nM T67619 CH14KD 23647018 IC50 = 21670 nM T67619 CQ5Z0J 23647019 IC50 > 50000 nM T67619 CT7XW8 23647020 IC50 = 3136 nM T67619 CG6D4M 23647319 IC50 > 10000 nM T67619 CY8Z7X 23647330 IC50 > 10000 nM T67619 C4XD8H 23647348 IC50 > 10000 nM T67619 CC26BS 23647380 IC50 = 0.34 nM T67619 C45OPN 23647431 IC50 = 1 nM T67619 CW7A4C 23647432 IC50 = 1.8 nM T67619 CL7V6D 23647433 IC50 = 953 nM T67619 C4W2MD 23647434 IC50 = 51 nM T67619 CGK64O 23647435 IC50 = 7.1 nM T67619 CK7SN2 23647436 IC50 = 223 nM T67619 CLX3Y0 23647437 IC50 = 14 nM T67619 CU5M4I 23647438 IC50 = 59 nM T67619 CRH7L6 23647439 IC50 = 104 nM T67619 CGC1Y2 23647440 IC50 = 13 nM T67619 CMO3B9 23647441 IC50 = 6.1 nM T67619 C1YH6X 23647442 IC50 = 228 nM T67619 C2V6RK 23647443 IC50 = 8.3 nM T67619 CKS3V6 23647541 IC50 = 7.4 nM T67619 CHCE50 23647542 IC50 = 5.4 nM T67619 C4VZB9 23647547 IC50 = 4.3 nM T67619 CI6VW5 23647548 IC50 = 99 nM T67619 C1ET9C 23647551 IC50 = 4 nM T67619 C1SQ4V 23647552 IC50 = 52.7 nM T67619 CK8OY5 23647554 IC50 = 80 nM T67619 C7RNQ4 23647555 IC50 = 1.5 nM T67619 CK60WI 23647570 IC50 = 4.6 nM T67619 C6PXR2 23647571 IC50 = 2 nM T67619 CRUN54 23647572 IC50 = 1.5 nM T67619 C2JTA3 23647573 IC50 = 0.8 nM T67619 C16RZH 23647574 IC50 = 1240 nM T67619 C3F5WY 23647575 IC50 = 84 nM T67619 CF57LO 23647576 IC50 = 697 nM T67619 C98UNX 23647577 IC50 = 227 nM T67619 CG2AS0 23647578 IC50 = 778 nM T67619 CZNA28 23647579 IC50 = 39500 nM T67619 CS7IQ0 23647580 IC50 = 160 nM T67619 C17HUI 23647581 IC50 = 3.5 nM T67619 CB0A3U 23647582 IC50 = 640 nM T67619 C5IN1M 23647583 IC50 = 144 nM T67619 C4FL0E 23647584 IC50 = 22 nM T67619 C03ZRM 23647585 IC50 = 57 nM T67619 CJO5X4 23647586 IC50 = 305 nM T67619 CWSE92 23647587 IC50 = 122 nM T67619 CS2LZ5 23647588 IC50 = 180 nM T67619 CTGH98 23647589 IC50 = 56 nM T67619 CYM86G 23647590 IC50 = 15 nM T67619 C2G1QI 23647591 IC50 = 995 nM T67619 CWI63J 23649242 IC50 = 176 nM T67619 CHI9J4 23654066 IC50 = 3315 nM T67619 C4KT2G 23654071 IC50 = 8 nM T67619 C3JWK1 23654166 IC50 = 18.3 nM T67619 CV8I2B 23654167 IC50 = 27 nM T67619 CU1M0Q 23654255 IC50 = 613 nM T67619 C8N4DL 23654256 IC50 > 3000 nM T67619 CDON60 23654258 IC50 = 453 nM T67619 CY7P0K 23654341 IC50 = 2406 nM T67619 C35HDM 23654345 IC50 = 15.4 nM T67619 C4TOU0 23654594 IC50 = 11.6 nM T67619 CG03YM 23654922 IC50 = 4.9 nM T67619 CL8M1D 23658126 IC50 > 50 nM T67619 C2RV3U 24180608 IC50 > 30000 nM T67619 C7YG1N 24759534 IC50 = 24000 nM T67619 CAJ4T2 24762205 IC50 > 10000 nM T67619 CQNP54 24764449 IC50 = 10000 nM T67619 CCPS81 24764502 IC50 > 35000 nM T67619 C4Z9CN 24769780 IC50 > 100000 nM T67619 CJUK39 24770517 IC50 > 10000 nM T67619 C0EKO5 24772654 IC50 > 10000 nM T67619 CW3JR8 24783593 IC50 = 4 nM T67619 C05MQY 24783594 IC50 = 901 nM T67619 C93TIM 24786152 IC50 = 6 nM T67619 CSY9Z6 24788164 IC50 = 196 nM T67619 CFR62V 24788432 IC50 = 5 nM T67619 C2JNI3 24788623 IC50 = 8 nM T67619 CMR7F1 24788739 IC50 = 5 nM T67619 CNZ1V8 24798741 IC50 = 151 nM T67619 CR1DI7 24798742 IC50 = 42 nM T67619 CP16TG 24802788 IC50 = 8 nM T67619 CN2IY6 24802961 IC50 = 25 nM T67619 CC1V3Y 24803300 IC50 = 63 nM T67619 C1FA4Y 24803301 IC50 = 63 nM T67619 CTM7N5 24803303 IC50 = 6 nM T67619 CY1ZS7 24803305 Ki = 0.06 nM T67619 CFJ87E 24803786 IC50 = 100 nM T67619 CRP87A 24803787 IC50 = 50 nM T67619 CYOS32 24803956 IC50 = 8 nM T67619 CJZ1Q9 24803957 IC50 = 40 nM T67619 C9YD5V 24803959 IC50 = 250 nM T67619 C3H4SB 24804133 IC50 = 2 nM T67619 C2ANO6 24804134 Ki = 0.04 nM T67619 CCD9R0 24804298 IC50 = 10 nM T67619 CO1HE7 24804299 IC50 = 4 nM T67619 CSH8A5 24804780 Ki = 0.79 nM T67619 CDTV63 24805106 IC50 = 3 nM T67619 CFL2N5 24805271 IC50 = 6 nM T67619 C2ZBE6 24805272 IC50 = 40 nM T67619 CUTH13 24805273 IC50 = 8 nM T67619 CQ3D0U 24805274 IC50 = 3 nM T67619 C8YZ2U 24805275 IC50 = 25 nM T67619 CHLM50 24805277 IC50 = 16 nM T67619 C9PA0M 24807809 IC50 > 30000 nM T67619 CQJ6I5 24814874 IC50 = 12000 nM T67619 CCP2M3 24822704 IC50 > 50000 nM T67619 CSW5V3 24865437 IC50 > 100000 nM T67619 CFK2B9 24882503 IC50 > 10000 nM T67619 C43HWQ 24883287 IC50 > 10000 nM T67619 C8DA5Q 24883334 IC50 > 10000 nM T67619 CW75GN 24889248 IC50 = 6 nM T67619 CGNT83 24889250 IC50 = 995 nM T67619 CWXY34 24889587 IC50 = 3 nM T67619 C5WS6R 24894100 IC50 = 13 nM T67619 CY8L7E 24896769 IC50 > 10000 nM T67619 CN13JF 24899915 IC50 > 10 ug.mL-1 T67619 CBWR97 24899916 IC50 = 5.3 ug.mL-1 T67619 C9F2JD 24899917 IC50 > 10 ug.mL-1 T67619 C64MTI 24900160 IC50 > 10 ug.mL-1 T67619 CO2I6Q 24900161 IC50 > 10 ug.mL-1 T67619 CP06SO 24949134 IC50 = 260 nM T67619 CXW60I 24949292 IC50 = 2468 nM T67619 C8UGZ5 24949295 IC50 = 1 nM T67619 CD04RG 24949296 IC50 = 11 nM T67619 C4SJ6L 24949446 IC50 = 4 nM T67619 C2YFP6 24949606 IC50 = 310 nM T67619 C9B0OX 24949764 IC50 = 22 nM T67619 C1KLG7 24949923 IC50 = 1201 nM T67619 CLZ23U 24951610 IC50 = 4800 nM T67619 CV5IE4 24963049 Ki = 0.2 nM T67619 CD5HQ0 24969301 IC50 > 10000 nM T67619 CC9LQ7 24971375 IC50 = 210 nM T67619 CE6S1A 24971376 IC50 > 10000 nM T67619 C69IYD 24971377 IC50 = 425 nM T67619 CM3AC2 24971378 IC50 = 318 nM T67619 CL78NU 24971379 IC50 = 171 nM T67619 C6R4UE 24971380 IC50 > 10000 nM T67619 CMY86O 24971381 IC50 = 294 nM T67619 C8FLD6 24971382 IC50 = 12.7 nM T67619 CTR3Q0 24971383 IC50 = 2790 nM T67619 C7HRA0 24971384 IC50 = 3190 nM T67619 C3DX1P 24971385 IC50 = 1330 nM T67619 CLJ2N0 24971386 IC50 = 226 nM T67619 CC7B8W 24971387 IC50 = 139 nM T67619 CCWV70 24971388 IC50 = 198 nM T67619 CSE34D 24971389 IC50 = 90 nM T67619 C5NFP2 24971390 IC50 = 137 nM T67619 C0B9HE 24971391 IC50 = 1521 nM T67619 CX1U6V 24971392 IC50 = 162 nM T67619 C3JT8Q 24971393 IC50 = 63 nM T67619 C4EG8R 24993189 IC50 > 10000 nM T67619 CA9F3Y 25023714 IC50 = 79 nM T67619 C8Z4PI 25023715 IC50 = 126 nM T67619 CV96QX 25023716 IC50 = 331 nM T67619 C5INV4 25023717 IC50 = 501 nM T67619 CPOH02 25023718 IC50 = 631 nM T67619 C6F7RD 25023719 IC50 = 562 nM T67619 CW2MV8 25023720 IC50 = 32 nM T67619 CPB4S2 25023721 IC50 = 79 nM T67619 C8UL4O 25023722 IC50 = 2760 nM T67619 CZ05HU 25023723 IC50 = 3160 nM T67619 CSM1R7 25023724 IC50 = 79 nM T67619 C4DF8X 25023725 IC50 = 1050 nM T67619 CXFQ18 25023726 IC50 = 1130 nM T67619 C13MHS 25023727 IC50 = 50 nM T67619 C1JEU6 25023729 IC50 = 9 nM T67619 C14NAT 25023731 IC50 = 2 nM T67619 C81XKW 25023732 IC50 = 3 nM T67619 CFH80B 25023733 IC50 = 1010 nM T67619 CR8JP7 25023735 IC50 = 400 nM T67619 C4W7LY 25023736 IC50 = 5 nM T67619 CA6QU5 25023737 IC50 = 3 nM T67619 CB7VT5 25032306 IC50 = 5.82 nM T67619 C2H3WJ 25032388 IC50 = 19.3 nM T67619 C17PCM 25032389 IC50 = 148 nM T67619 CM1GB6 25032390 IC50 = 376 nM T67619 C0W2TF 25032391 IC50 = 51.9 nM T67619 CCR6S7 25032392 IC50 = 56.8 nM T67619 CX1HL8 25032704 Ki > 8210 nM T67619 CL7V8R 25060409 IC50 = 377 nM T67619 CFU5E2 25060410 IC50 = 712 nM T67619 C3B8FI 25060411 IC50 = 78 nM T67619 C4CJX9 25060675 IC50 = 889 nM T67619 COV3Q4 25061501 IC50 = 0.5 nM T67619 C6P1CX 25066843 IC50 > 20000 nM T67619 CM07IN 25093232 IC50 = 6436 nM T67619 CV42JO 25093234 IC50 = 8819 nM T67619 CIH3E5 25093235 IC50 = 7491 nM T67619 C2KY1G 25094210 IC50 > 10000 nM T67619 C6BWZ8 25145145 IC50 > 100 nM T67619 C78YWA 25145716 IC50 > 500 nM T67619 CCK8D2 25154767 IC50 > 20000 nM T67619 C3FQO6 25156555 IC50 = 14000 nM T67619 CTM0J8 25156556 IC50 = 17000 nM T67619 C8NR9H 25170562 IC50 = 241 nM T67619 CS9LC3 25170563 IC50 = 530 nM T67619 CN8YZ4 25170991 IC50 = 12 nM T67619 CNJH95 25175218 IC50 = 85 nM T67619 C53JCN 25175220 IC50 = 1600 nM T67619 CIG4H0 25178539 IC50 = 9000 nM T67619 CX8F3W 25183032 IC50 > 5000 nM T67619 C2DFB6 25189112 IC50 = 150 nM T67619 CK2XD0 25189383 IC50 = 163 nM T67619 CHN5O0 25190977 IC50 = 1 nM T67619 CNG96H 25210579 IC50 > 10000 nM T67619 CRO09K 25211064 IC50 > 30000 nM T67619 COWB90 25221040 IC50 = 6 nM T67619 CC25TV 25222706 IC50 = 1 nM T67619 C1IG7E 25243798 IC50 = 28 nM T67619 CH65JV 25243799 IC50 = 2.8 nM T67619 CDR19S 25243801 IC50 = 22000 nM T67619 C7BAN0 25262260 IC50 > 20000 nM T67619 CBQO98 42602095 IC50 = 8 nM T67619 CJ61SE 42602096 IC50 = 7 nM T67619 CI42XG 42602097 IC50 = 5 nM T67619 CD2AH4 42602175 IC50 = 6 nM T67619 CSWA85 42602176 IC50 = 7 nM T67619 C1LUN4 42602178 IC50 = 2 nM T67619 C8O3EA 42602260 IC50 = 4 nM T67619 C93NKL 42602264 IC50 = 3 nM T67619 C7WPJ5 42602351 IC50 = 12 nM T67619 CI2EM9 42612826 IC50 = 99 nM T67619 CWS37O 42618140 IC50 = 5011.87 nM T67619 C2JV3O 42618143 IC50 > 10000 nM T67619 CG01BO 42618144 IC50 > 10000 nM T67619 C8JRS9 42618236 IC50 = 497 nM T67619 CM8JE5 42618237 IC50 = 44 nM T67619 CV6WU1 42618238 IC50 = 57 nM T67619 C5TWM3 42618240 IC50 = 80 nM T67619 CCS6L2 42618243 IC50 = 295 nM T67619 C50WPV 42618244 IC50 = 350 nM T67619 CX1M5O 42618245 IC50 = 383 nM T67619 C02GUX 42618246 IC50 = 850 nM T67619 C18ILO 42618247 IC50 = 1440 nM T67619 C8B0CI 42625066 IC50 = 72 nM T67619 CJ5U1X 42639664 IC50 > 10 ug.mL-1 T67619 C5IDL4 44123827 IC50 = 19000 nM T67619 C3ROX1 44124863 IC50 = 13 nM T67619 C2YQX8 44125256 IC50 = 415 nM T67619 CV5O8L 44125375 IC50 = 335 nM T67619 C5JN4O 44125376 IC50 > 12000 nM T67619 C0U2OY 44125377 IC50 = 118 nM T67619 C0HB4C 44129168 IC50 = 5000 nM T67619 CLW80F 44160269 IC50 = 2400 nM T67619 CYN65S 44205558 IC50 = 85900 nM T67619 CK73NR 44219749 IC50 > 50000 nM T67619 C59CDG 44389260 IC50 = 273 nM T67619 CSBC59 44396134 IC50 > 20000 nM T67619 CGI5L7 44405938 IC50 > 20000 nM T67619 C0G3WF 44405939 IC50 > 20000 nM T67619 CR3Q7Z 44405940 IC50 > 20000 nM T67619 C79WRL 44405941 IC50 > 20000 nM T67619 C9ZNA0 44405945 IC50 > 100000 nM T67619 C9LD2T 44405946 IC50 > 100000 nM T67619 C0RO6U 44405949 IC50 = 9000 nM T67619 C2CTN7 44405982 IC50 > 100000 nM T67619 C0CR1O 44405983 IC50 = 16000 nM T67619 CW86VI 44405987 IC50 > 100000 nM T67619 C5V4TQ 44405999 IC50 > 100000 nM T67619 C0XZ8K 44406013 IC50 > 20000 nM T67619 CS3K1P 44406014 IC50 > 20000 nM T67619 CC93JP 44406018 IC50 > 20000 nM T67619 C7P0IH 44406019 IC50 > 20000 nM T67619 C4X2ME 44406047 IC50 > 100000 nM T67619 C36YDV 44406048 IC50 > 100000 nM T67619 CXZ5C3 44406055 IC50 = 17000 nM T67619 CCRZ12 44406074 IC50 > 20000 nM T67619 C7LOE3 44412808 IC50 = 5.4 nM T67619 C7EB4A 44412822 IC50 = 488 nM T67619 CQ9G6N 44412832 IC50 = 7.2 nM T67619 CMF8W1 44412836 IC50 = 41 nM T67619 C3N5EC 44412847 IC50 = 0.9 nM T67619 CR7OD4 44412850 IC50 = 4400 nM T67619 CN0L7F 44412860 IC50 = 2500 nM T67619 CBS2H9 44412862 IC50 = 3.2 nM T67619 C61OIQ 44412873 IC50 = 0.7 nM T67619 C0N8HB 44412905 IC50 = 7.4 nM T67619 CX69NO 44412915 IC50 = 1.5 nM T67619 CNS6T5 44412926 IC50 = 4.3 nM T67619 C4Y1SK 44412938 IC50 = 660 nM T67619 CP1X0H 44412967 IC50 = 352 nM T67619 CY91EG 44412972 IC50 = 3.3 nM T67619 CI5TM8 44412973 IC50 = 8.2 nM T67619 CU3OI4 44412985 IC50 = 179 nM T67619 CF90ZW 44412987 IC50 = 405 nM T67619 CDQ27J 44412995 IC50 = 5.9 nM T67619 C8IHO0 44412996 IC50 = 1.2 nM T67619 CC32EP 44412997 IC50 = 153 nM T67619 CPR4A0 44413008 IC50 = 10.4 nM T67619 C2OB6S 44413011 IC50 = 99 nM T67619 CF3XQ7 44413017 IC50 = 10.3 nM T67619 CRM74H 44413021 IC50 = 147 nM T67619 CM4VS2 44413034 IC50 = 20700 nM T67619 C32AGE 44413035 IC50 = 15600 nM T67619 COT37A 44413036 IC50 = 24.6 nM T67619 CLA2M5 44413047 IC50 = 40.3 nM T67619 CVR6J9 44413051 IC50 = 4 nM T67619 CK2OF4 44413052 IC50 = 80 nM T67619 C1W3QV 44413053 IC50 = 1020 nM T67619 C7T8CS 44413054 IC50 = 52.7 nM T67619 CT5DW8 44413055 IC50 = 1.5 nM T67619 CKEJ69 44413061 IC50 = 10 nM T67619 CG3M5B 44420151 IC50 = 15800 nM T67619 CUBS93 44420157 IC50 > 50000 nM T67619 C87IEZ 44420158 IC50 > 50000 nM T67619 C3U6EZ 44420161 IC50 = 16000 nM T67619 C69FMK 44420162 IC50 = 4900 nM T67619 C93WSL 44420163 IC50 = 12400 nM T67619 CWF80D 44420170 IC50 = 13900 nM T67619 C2PMR5 44420171 IC50 > 50000 nM T67619 CWVG37 44420172 IC50 = 12300 nM T67619 CETQ79 44427518 IC50 = 880 nM T67619 COPG94 44427519 IC50 > 10000 nM T67619 CRT01D 44440036 IC50 > 500000 nM T67619 C7BV9Y 44440046 IC50 > 500000 nM T67619 CZG58I 44440056 IC50 > 500000 nM T67619 CF1V2S 44440064 IC50 = 445000 nM T67619 C2C5PI 44440069 IC50 = 409000 nM T67619 CFB1Z9 44440071 IC50 = 241000 nM T67619 C7N9HX 44440091 IC50 = 229000 nM T67619 CI6G1H 44440096 IC50 = 239000 nM T67619 CZN6H8 44440098 IC50 = 438000 nM T67619 C9WFY1 44440102 IC50 = 28000 nM T67619 C08TXI 44440105 IC50 = 36000 nM T67619 CM92AD 44440107 IC50 = 52000 nM T67619 C6B1KJ 44440111 IC50 = 62000 nM T67619 C2CMA7 44440117 IC50 = 94000 nM T67619 CU1I5Y 44440122 IC50 = 96000 nM T67619 C0GL1Y 44440125 IC50 = 322000 nM T67619 CVMW10 44440127 IC50 > 500000 nM T67619 CFEW28 44440132 IC50 = 41000 nM T67619 CI95LP 44440133 IC50 = 79000 nM T67619 CZNU95 44440139 IC50 > 500000 nM T67619 C9A0SE 44440142 IC50 = 51000 nM T67619 C8CIM1 44440145 IC50 = 89000 nM T67619 CJ5LO1 44440146 IC50 = 104000 nM T67619 C8OFZ6 44440150 IC50 = 119000 nM T67619 CMC56G 44440151 IC50 = 163000 nM T67619 C4VI5W 44440153 IC50 = 193000 nM T67619 C4IG3K 44440154 IC50 = 390000 nM T67619 C8UOT2 44440155 IC50 = 77000 nM T67619 C2SA8C 44440158 IC50 > 500000 nM T67619 CN5P8W 44440160 IC50 = 120000 nM T67619 C6IJ5S 44440184 IC50 = 58000 nM T67619 CHP41T 44442415 IC50 = 41 nM T67619 CI26UX 44442416 IC50 = 15 nM T67619 C2W1RN 44442417 IC50 = 81 nM T67619 C4A9FD 44442418 IC50 = 24 nM T67619 COP8A3 44449880 IC50 = 3.5 nM T67619 CMC82Z 44449900 IC50 = 5.6 nM T67619 C3APO5 44449908 IC50 = 7.4 nM T67619 CA85HS 44449909 IC50 = 21 nM T67619 C4QJK8 44449942 IC50 = 470 nM T67619 C0ICB5 44449973 IC50 = 44 nM T67619 CE15WY 44449975 IC50 = 250 nM T67619 CEWB75 44450002 IC50 = 120 nM T67619 CDEJ84 44450004 IC50 = 75 nM T67619 CZ1R8M 44450033 IC50 > 100000 nM T67619 CIY3T5 44450035 IC50 > 100000 nM T67619 C5Y4PN 44450059 IC50 > 100000 nM T67619 C28LMV 44450060 IC50 > 100000 nM T67619 CC7O6L 44454395 IC50 = 139 nM T67619 C9ZML1 44454396 IC50 = 45 nM T67619 C8OG1V 44517709 IC50 = 2600 nM T67619 C94NTS 44555483 IC50 = 10000 nM T67619 C1EVH2 44560678 IC50 = 1408 nM T67619 CI58CZ 44560679 IC50 = 3.5 nM T67619 CC4Z5M 44560681 IC50 = 26 nM T67619 CWOM65 44560715 IC50 = 25 nM T67619 C7YCO3 44560716 IC50 = 37 nM T67619 C5X7PO 44560717 IC50 = 35 nM T67619 COTH35 44560718 IC50 = 20 nM T67619 C6J0ZC 44560719 IC50 = 38 nM T67619 CL0A2D 44560720 IC50 = 37 nM T67619 CR8K0X 44560724 IC50 = 88 nM T67619 CE08JD 44560725 IC50 = 67 nM T67619 CSX84T 44560726 IC50 = 18 nM T67619 C1O0IG 44560727 IC50 = 10 nM T67619 CB7X4S 44560728 IC50 = 52 nM T67619 C94LIO 44560729 IC50 = 72 nM T67619 C3UQ8C 44560730 IC50 = 104 nM T67619 C8OD4F 44560731 IC50 = 70 nM T67619 CLB20U 44560732 IC50 = 115 nM T67619 CGY1X7 44561054 IC50 = 43 nM T67619 CZK43G 44561055 IC50 = 208 nM T67619 C4WLX8 44561056 IC50 = 25 nM T67619 CXC8I3 44561057 IC50 = 7 nM T67619 CS0QZ4 44561058 IC50 = 285 nM T67619 C1QG9P 44561059 IC50 = 720 nM T67619 C9MTS4 44561060 IC50 = 924 nM T67619 CKV96M 44571730 IC50 > 20000 nM T67619 CZ9L8F 44572052 IC50 = 265.5 nM T67619 CIV48S 44572053 IC50 = 26.7 nM T67619 CFVA91 44572054 IC50 = 9.9 nM T67619 CZE8M9 44572055 IC50 = 41.8 nM T67619 CT0R7C 44581248 IC50 = 2.5 nM T67619 C89HYP 44588980 IC50 = 1410 nM T67619 C2J9RS 44590344 IC50 = 78000 nM T67619 CKCR57 44590345 IC50 = 50000 nM T67619 CXJG68 44590346 IC50 > 500000 nM T67619 C3XFW2 44590347 IC50 = 16000 nM T67619 CK1MU5 44590348 IC50 = 78000 nM T67619 CWG8H9 44590349 IC50 = 288000 nM T67619 C51SAK 44590350 IC50 = 173000 nM T67619 CP3V1F 44590351 IC50 = 96000 nM T67619 CR8I2S 44590352 IC50 = 84000 nM T67619 CZ1AX7 44590353 IC50 = 215000 nM T67619 C5F3MT 44590354 IC50 = 152000 nM T67619 C3WJ5A 44590355 IC50 = 84000 nM T67619 CL7K6O 44590356 IC50 = 55000 nM T67619 C0S3TK 44590357 IC50 = 43000 nM T67619 CN7R1H 44590358 IC50 = 28000 nM T67619 CGUM97 44590359 IC50 = 23000 nM T67619 C9ISJ4 44590360 IC50 = 38000 nM T67619 CL82MA 44590361 IC50 = 17000 nM T67619 C7YT2M 44590362 IC50 = 253000 nM T67619 C6MK9B 44590363 IC50 = 158000 nM T67619 CLKF87 44590364 IC50 = 83000 nM T67619 C2ML8U 44590365 IC50 = 52000 nM T67619 C58ETF 44590366 IC50 = 44000 nM T67619 CQ52SV 44590405 IC50 = 126000 nM T67619 C4KS7X 44590406 IC50 = 32000 nM T67619 CJG86C 44590407 IC50 = 112000 nM T67619 CWP69C 44590408 IC50 = 232000 nM T67619 C0DJS1 44591843 Ki = 0.05 nM T67619 CX52YW 44591844 Ki = 0.1 nM T67619 C1LS6V 44591845 IC50 = 2 nM T67619 C2EMA5 44592331 IC50 = 158 nM T67619 CXK27N 44592363 IC50 = 20 nM T67619 C2W3NO 44592364 IC50 = 20 nM T67619 CSZ5R9 44592438 Ki = 20 nM T67619 C6X7FC 44592501 Ki = 2 nM T67619 CTS95L 44592502 IC50 = 3 nM T67619 CSKZ16 44592503 IC50 = 1 nM T67619 COY57J 44592504 Ki = 0.03 nM T67619 C3CDV8 44592505 Ki = 0.06 nM T67619 CVW08Q 44608012 IC50 = 261 nM T67619 C1SIK2 44620952 IC50 = 259 nM T67619 CAE82W 44623107 IC50 = 5 nM T67619 CNX84R 44817010 IC50 = 8500 nM T67619 C0U1IR 45139233 Ki = 260 nM T67619 CK49WN 45139234 Ki = 1100 nM T67619 CU3RF1 45139989 IC50 > 10000 nM T67619 CQGZ06 45139991 IC50 > 10000 nM T67619 CQ7OZ9 45142021 IC50 = 3.8 nM T67619 CU2K8B 45142026 IC50 = 4.2 nM T67619 CLCU70 45142256 IC50 = 7.2 nM T67619 C1V2YL 45142259 IC50 = 6.5 nM T67619 CIGO65 45480169 IC50 = 180 nM T67619 C9K3BG 45481616 IC50 = 0.8 nM T67619 CM3J5L 45481618 IC50 = 312 nM T67619 CC10HR 45481731 IC50 = 1848 nM T67619 CG1CH8 45481732 IC50 = 1360 nM T67619 C6RGK5 45481733 IC50 = 2020 nM T67619 C81MPU 45481734 IC50 = 47 nM T67619 C7E5QJ 45481735 IC50 = 65.5 nM T67619 C05ULY 45481736 IC50 = 8.4 nM T67619 C1GT9Y 45481737 IC50 = 39 nM T67619 C4E7GT 45481738 IC50 = 18 nM T67619 CLV13D 45481739 IC50 = 14 nM T67619 CF92RB 45481740 IC50 = 12 nM T67619 CUDW68 45481741 IC50 = 5 nM T67619 C4C1UM 45481742 IC50 = 3.9 nM T67619 CHL24S 45481743 IC50 = 2.5 nM T67619 C6HXS1 45481744 IC50 = 6 nM T67619 CWLJ43 45481745 IC50 = 751 nM T67619 C5TM4L 45481746 IC50 = 6.8 nM T67619 CRC95S 45481747 IC50 = 210 nM T67619 CN4M9E 45482050 IC50 = 1.4 nM T67619 CZ5XQ0 45482051 IC50 = 8.2 nM T67619 C9CB5D 45482052 IC50 = 1120 nM T67619 C21CBP 45482053 IC50 = 7.2 nM T67619 CX7M1A 45482054 IC50 = 3.3 nM T67619 CAM5B6 45482055 IC50 = 40.3 nM T67619 C1RHW8 45482056 IC50 = 153 nM T67619 C05RJC 45482057 IC50 = 0.17 nM T67619 C75SVJ 45482058 IC50 = 5.9 nM T67619 C9X1AB 45482059 IC50 = 10.4 nM T67619 C4L8WS 45482060 IC50 = 10.3 nM T67619 CX5Y2C 45482061 IC50 = 1.5 nM T67619 C3FO0V 45482457 IC50 = 760 nM T67619 CX14WY 45482459 IC50 = 63 nM T67619 C2YB4R 45482460 IC50 = 20 nM T67619 C96GDA 45482461 IC50 = 1089 nM T67619 CK2O4Z 45482463 IC50 = 16000 nM T67619 CJ4V8P 45482465 IC50 = 12300 nM T67619 CH46FZ 45482466 IC50 = 0.9 nM T67619 CCL20J 45482467 IC50 = 0.7 nM T67619 C6VCU9 45482468 IC50 = 21200 nM T67619 CTP1O0 45482469 IC50 = 10 nM T67619 CASO36 46182743 IC50 = 14.3 nM T67619 C4CBT9 46190874 IC50 = 0.8 nM T67619 CH9I5S 46190875 IC50 = 1 nM T67619 CQ5SD4 46190876 IC50 = 2 nM T67619 CQYO76 46192856 IC50 = 402 nM T67619 CU1Q0K 46192857 IC50 = 422 nM T67619 CQ82JV 46192858 IC50 = 318 nM T67619 CN0A1I 46192859 IC50 = 905 nM T67619 CM96WL 46192860 IC50 = 1395 nM T67619 CDJS49 46192989 IC50 = 183 nM T67619 CS9T2M 46192991 IC50 = 251 nM T67619 CD4O0S 46192992 IC50 = 209 nM T67619 CPK5N7 46193129 IC50 = 302 nM T67619 CQ8YW5 46193130 IC50 = 1324 nM T67619 C3VYA4 46193131 IC50 = 793 nM T67619 CS5Q2R 46193132 IC50 = 433 nM T67619 C52HOD 46193133 IC50 = 1750 nM T67619 CF57GK 46215462 IC50 > 10000 nM T67619 CZ58FY 46215814 IC50 > 10000 nM T67619 CY3HW5 46224684 IC50 = 1000 nM T67619 C1J6GR 46224908 IC50 > 10000 nM T67619 CSWY60 46225572 IC50 = 1 nM T67619 CS9GL5 46225573 IC50 = 12 nM T67619 CB5H9C 46225574 IC50 = 1 nM T67619 C8M1DT 46225589 IC50 = 1 nM T67619 CZ70MO 46226075 IC50 = 0.8 nM T67619 CC82WK 46226076 IC50 = 1 nM T67619 CQVW97 46226077 IC50 = 8 nM T67619 CYW1K4 46226078 IC50 = 13 nM T67619 C60XUQ 46226079 IC50 = 3 nM T67619 C5PCH8 46226080 IC50 = 1 nM T67619 CIX07W 46226091 IC50 = 10 nM T67619 C6UD1Y 46226095 IC50 = 10 nM T67619 C7IF4T 46226096 IC50 = 3 nM T67619 CUDZ46 46226135 IC50 = 500 nM T67619 C0P4CT 46226136 IC50 = 1 nM T67619 CPH49S 46226137 IC50 = 1 nM T67619 CM5X8B 46226156 IC50 = 1 nM T67619 CGA0E5 46226413 IC50 = 50 nM T67619 CLW06M 46226414 IC50 = 10500 nM T67619 C64TVL 46226417 IC50 = 1 nM T67619 CI90DE 46226435 IC50 = 720 nM T67619 CHD02B 46226697 IC50 > 50000 nM T67619 CJZA45 46232267 IC50 > 100000 nM T67619 C3PLE6 46232269 IC50 > 100000 nM T67619 C3U8HV 46232270 IC50 > 100000 nM T67619 CYA73D 46232312 IC50 > 100000 nM T67619 CYT37A 46232443 IC50 > 50000 nM T67619 C48ZVW 46232555 IC50 > 50000 nM T67619 CS9B1U 46232556 IC50 > 50000 nM T67619 CC2WT4 46232590 IC50 = 11400 nM T67619 C7ON5A 46233287 IC50 > 10000 nM T67619 CC0L3B 46837499 IC50 = 68 nM T67619 C73KIU 46837500 IC50 = 200 nM T67619 CZ40RT 46837624 IC50 = 4 nM T67619 C5B1AE 46837625 IC50 = 10000 nM T67619 CD5NX6 46837626 IC50 = 700 nM T67619 CT68HQ 46837627 IC50 = 4000 nM T67619 C3W7VO 46837628 IC50 = 600 nM T67619 CUS83Q 46837629 IC50 = 700 nM T67619 CUL02J 46837630 IC50 = 1900 nM T67619 CAQ80P 46837631 IC50 = 2400 nM T67619 CBN65Q 46837763 IC50 = 56 nM T67619 C6SDE5 46837764 IC50 = 765 nM T67619 CH93TZ 46837765 IC50 = 58 nM T67619 CC5NB6 46837766 IC50 = 61 nM T67619 C3Q2LA 46837768 IC50 = 16 nM T67619 C61OYM 46837903 IC50 = 62 nM T67619 CWP9G3 46837904 IC50 = 44 nM T67619 C31BZG 46837905 IC50 = 38 nM T67619 CTO76L 46837906 IC50 = 7.4 nM T67619 CYT5C1 46837907 IC50 = 7.8 nM T67619 C4VO3C 46837908 IC50 = 3 nM T67619 CHZ86X 46838046 IC50 = 2.6 nM T67619 CL9P5G 46838047 IC50 = 1.4 nM T67619 CI3K7B 46838048 IC50 = 17.5 nM T67619 C65KZS 46838049 IC50 = 11.4 nM T67619 CU8FG3 46838050 IC50 = 3.3 nM T67619 CTLO06 46838051 IC50 = 1.8 nM T67619 C68OGL 46838189 IC50 = 7.7 nM T67619 CXVB91 46838190 IC50 = 1 nM T67619 CSNU98 46838191 IC50 = 1.1 nM T67619 COTJ39 46863083 IC50 > 30000 nM T67619 C7H4YM 46865419 IC50 > 10000 nM T67619 CD57BJ 46870040 IC50 = 5 nM T67619 CLS29B 46872626 IC50 > 10000 nM T67619 C9WY0Q 46880284 IC50 = 491 nM T67619 C9CKW4 46880292 IC50 = 404 nM T67619 CROD39 46880293 IC50 = 17 nM T67619 CE1J3N 46880294 IC50 = 40 nM T67619 C8XRP1 46880324 IC50 = 370 nM T67619 CE8HO7 46880330 IC50 = 35 nM T67619 CA23RZ 46880364 IC50 = 181 nM T67619 CJT92P 46880365 IC50 = 413 nM T67619 CNQ6Y4 46880366 IC50 = 368 nM T67619 CLQ62J 46880370 IC50 = 141 nM T67619 C2U9SD 46880371 IC50 = 895 nM T67619 CSYB29 46880407 IC50 = 280 nM T67619 C49KDO 46880415 IC50 = 8.5 nM T67619 CMW01F 46880416 IC50 = 77 nM T67619 CW7OT8 46880504 IC50 > 1000 nM T67619 C37GCR 46880505 IC50 = 95 nM T67619 CJ1B8S 46880932 IC50 = 76 nM T67619 CF1BM3 46880933 IC50 > 2200 nM T67619 C9TLK1 46880934 IC50 = 198 nM T67619 CTD7W6 46886255 IC50 = 940 nM T67619 CXJ92T 46886273 IC50 = 840 nM T67619 CRU26Y 46886274 IC50 = 1170 nM T67619 C5UJN8 46886283 IC50 = 920 nM T67619 C9FN2O 46886284 IC50 = 2030 nM T67619 COC48H 46886291 IC50 = 400 nM T67619 CM8RX4 46886549 Ki = 3 nM T67619 C70BLN 46886550 Ki = 1.9 nM T67619 CCV96R 46886665 IC50 = 5 nM T67619 C60GAV 46929544 IC50 > 8000 nM T67619 CP34VL 46929748 IC50 > 1000 nM T67619 CJ2E9Q 46929857 IC50 > 25000 nM T67619 C7AHF2 46942379 IC50 = 3629 nM T67619 C7F2NZ 46945659 IC50 = 3 nM T67619 CO94GU 46945660 IC50 = 8 nM T67619 CANS92 46945661 IC50 = 5 nM T67619 C2B5XF 49765254 IC50 > 10000 nM T67619 C9K1XO 49800133 IC50 = 5.7 nM T67619 C3D2RG 49800134 IC50 = 5.74 nM T67619 CQ93PT 49800135 IC50 = 25 nM T67619 CWI3E0 49800136 IC50 = 68 nM T67619 CHSF07 49806372 IC50 > 1000 nM T67619 C5ME3S 49806721 IC50 > 50000 nM T67619 CJZ5A0 49840306 IC50 > 10000 nM T67619 CF91RS 49843531 IC50 > 10000 nM T67619 COLG92 49860221 IC50 = 4 nM T67619 C9Z2EQ 49860222 IC50 = 3000 nM T67619 CH3E7S 49860227 IC50 = 355 nM T67619 C0DRX5 50898538 IC50 = 30000 nM T67619 C2Y6QS 50938552 IC50 > 10000 nM T67619 CKY3V1 50990924 IC50 = 6.3 nM T67619 CAZQ43 51003133 IC50 > 1000 nM T67619 C9NYP4 51036677 IC50 > 10000 nM T67619 C4WRY3 51037112 IC50 > 10000 nM T67619 CRI28Z 51037948 IC50 > 10000 nM T67619 C8CGM9 51346966 IC50 = 5 nM T67619 C73ANH 51353707 IC50 = 2500 nM T67619 CI4A6R 51353708 IC50 = 336 nM T67619 CJ4ZL6 51353709 IC50 = 305 nM T67619 CDLF71 51353710 IC50 = 4010 nM T67619 C04EVK 51353711 IC50 = 676 nM T67619 CD6AL8 51353712 IC50 > 5000 nM T67619 CPQ1G6 51354021 IC50 > 5000 nM T67619 CVK95R 51354022 IC50 = 1260 nM T67619 CHKA96 51354023 IC50 = 334 nM T67619 C6VD0B 51354313 IC50 = 33 nM T67619 CJC90Y 51354315 IC50 = 103 nM T67619 COH9L7 51354317 IC50 = 739 nM T67619 CV6I5D 51354595 IC50 = 1160 nM T67619 C1V6RN 51354597 IC50 = 757 nM T67619 CZ32XV 51354599 IC50 = 18 nM T67619 C8WEN4 51354600 IC50 = 5 nM T67619 C76KOV 51354878 IC50 = 8 nM T67619 CA3O2L 51354879 IC50 = 12 nM T67619 C0O2PW 51354880 IC50 = 19 nM T67619 C3JV4L 51354881 IC50 = 4.9 nM T67619 C6NL1Z 51354882 IC50 = 12 nM T67619 CPWD73 51354883 IC50 = 8.7 nM T67619 CB10AP 51355171 IC50 = 13 nM T67619 CKE42Q 51355172 IC50 = 7 nM T67619 CZF89J 51355173 IC50 = 9 nM T67619 CQF0J9 51355174 IC50 = 13 nM T67619 CI7MJ6 51357948 IC50 = 2800 nM T67619 C3B2KJ 52918145 IC50 = 19 nM T67619 C1AH3S 52918146 IC50 = 4 nM T67619 CVI2X4 52918147 IC50 = 3 nM T67619 C3X6JB 52918286 IC50 = 40 nM T67619 CXA03W 52920796 IC50 > 100 nM T67619 CEQN27 52936621 Ki > 1000 nM T67619 CM24LF 52938983 IC50 = 4.72 nM T67619 CMB47R 52940747 IC50 = 98 nM T67619 C4TUP9 52940786 IC50 = 868 nM T67619 CC1Y0M 52941299 IC50 = 838 nM T67619 CE73VJ 52941439 IC50 = 22920 nM T67619 CDT94U 52941495 IC50 = 150 nM T67619 CK7B9D 52941544 IC50 = 1 nM T67619 C9UF6K 52941555 IC50 = 51 nM T67619 CGQ9D4 52941556 IC50 = 2 nM T67619 CYM80Q 52942489 IC50 = 2883 nM T67619 CS09YT 52942516 IC50 = 690 nM T67619 C7G1KY 52942566 IC50 = 2 nM T67619 CJ4PF1 52942590 IC50 = 3321 nM T67619 CDF46K 52942649 IC50 = 80 nM T67619 CQ08WT 52942668 IC50 = 118 nM T67619 CJ3X1P 52942736 IC50 = 1 nM T67619 CM5Y2A 52943319 IC50 = 3203 nM T67619 CKCP18 52943685 IC50 = 88 nM T67619 CPO67Q 52943849 IC50 = 43 nM T67619 CHW04J 52943916 IC50 = 74 nM T67619 C1UYM2 52943963 IC50 = 2 nM T67619 CX7H0V 52944069 IC50 = 25000 nM T67619 CQ5IW7 52944431 IC50 = 809 nM T67619 CRL15Q 52944581 IC50 = 21233 nM T67619 CY8BV4 52944892 IC50 = 95 nM T67619 C86HVR 52944982 IC50 = 114 nM T67619 C2VOL8 52946136 IC50 = 30 nM T67619 CP1I6J 52946204 IC50 = 30 nM T67619 CFP7H2 52946232 IC50 = 2 nM T67619 CEM95A 52946401 IC50 = 595 nM T67619 CKE3C7 52946402 IC50 = 142 nM T67619 CFUA95 52946885 IC50 = 1460 nM T67619 CA80TG 52947050 IC50 = 25000 nM T67619 CXZA27 52947056 IC50 = 46 nM T67619 CDC98H 52947346 IC50 = 18 nM T67619 CXAP29 52947428 IC50 = 63 nM T67619 CTB27D 52947459 IC50 = 100 nM T67619 C8A1UQ 52947460 IC50 = 604 nM T67619 C3Q4CU 52947490 IC50 = 884 nM T67619 CB0HK1 52947582 IC50 = 104 nM T67619 CR9E1Z 52947590 IC50 = 2346 nM T67619 CQGI45 52947670 IC50 = 160 nM T67619 CB31ES 52948681 IC50 = 54 nM T67619 C5T7NA 52948731 IC50 = 8122 nM T67619 CK27CL 52948802 IC50 = 2 nM T67619 C50YOB 52949258 IC50 = 536 nM T67619 CKZ2N3 52949939 IC50 = 2048 nM T67619 CE81HA 52950003 IC50 = 30 nM T67619 C3TU8R 52950063 IC50 = 81 nM T67619 C7MC5G 52950205 IC50 = 284 nM T67619 C6OTY5 53251320 IC50 = 16000 nM T67619 CWV91D 53262404 IC50 = 5.4 nM T67619 C0KPF8 53316665 IC50 = 137 nM T67619 CE8OY2 53317913 IC50 > 100 nM T67619 CTK53X 53317972 IC50 = 92 nM T67619 C6EU4A 53318869 IC50 = 587 nM T67619 CWQX19 53319315 IC50 = 3 nM T67619 CDVB42 53321918 IC50 = 3 nM T67619 CJVR52 53324323 IC50 = 52 nM T67619 CQ6X4K 53324602 IC50 = 615 nM T67619 CP70YV 53325900 IC50 = 3 nM T67619 CR48EX 53325901 IC50 = 10 nM T67619 CM5Q3N 53325902 IC50 = 127 nM T67619 CBR4Q1 53325903 IC50 = 6 nM T67619 C62MCY 53325904 IC50 = 18 nM T67619 CJC4Y6 53326722 IC50 = 3 nM T67619 CF0XU9 53348197 IC50 = 9 nM T67619 C0SWH5 53348216 IC50 > 40000 nM T67619 CM7P3W 53357328 IC50 > 50000 nM T67619 CBPR36 53363353 IC50 = 769 nM T67619 C8NA4L 53384644 IC50 > 30000 nM T67619 C1CA4M 53386721 IC50 = 7 nM T67619 CW98EQ 53386722 IC50 = 390 nM T67619 CIA2K6 53386770 IC50 = 2150 nM T67619 C3O2YQ 53387086 IC50 = 320 nM T67619 C4X2NT 53387087 IC50 = 220 nM T67619 CHG4D7 53387088 IC50 = 320 nM T67619 C5H2OZ 53387248 IC50 = 250 nM T67619 CHZW84 53387249 IC50 = 130 nM T67619 CJG4C0 53387250 IC50 = 150 nM T67619 C2KP0Y 53387404 IC50 = 110 nM T67619 C4TWU9 53387405 IC50 = 176 nM T67619 CN2QM6 53387406 IC50 = 128 nM T67619 C5SMC3 53387410 IC50 = 50 nM T67619 C5Q0HA 53387411 IC50 = 574 nM T67619 CVS46X 53387568 IC50 = 130 nM T67619 C6DYT1 53387569 IC50 = 160 nM T67619 C90KZU 53387571 IC50 > 12000 nM T67619 CMO9K1 53387572 IC50 > 12000 nM T67619 CI40BG 53387573 IC50 = 101 nM T67619 C2IJR7 53387574 IC50 > 12000 nM T67619 CWB79U 53387575 IC50 > 12000 nM T67619 CB4H9G 53387738 IC50 = 1100 nM T67619 C5ZY9R 53387740 IC50 > 12000 nM T67619 C84SHL 53388204 IC50 = 282 nM T67619 CB5NA9 53388374 IC50 = 170 nM T67619 CQ6DV2 53388537 IC50 = 280 nM T67619 C1CB2R 53388538 IC50 = 290 nM T67619 CB1O3I 53388682 IC50 = 950 nM T67619 CMSX64 53388685 IC50 = 320 nM T67619 CXF90L 53388978 IC50 = 390 nM T67619 CLFK76 53389132 IC50 = 860 nM T67619 CQJ17T 53389133 IC50 = 240 nM T67619 CYU3W0 54580121 IC50 = 17 nM T67619 CC9W1Z 54580122 IC50 = 2400 nM T67619 C86YVW 54580123 IC50 = 250 nM T67619 CCS79P 54580124 IC50 = 9 nM T67619 C36VKO 54580125 IC50 = 17 nM T67619 CX5L3C 54580179 IC50 = 300 nM T67619 CCM46G 54580180 IC50 = 1100 nM T67619 CG7R6T 54580208 IC50 = 20000 nM T67619 C4O2KP 54580209 IC50 = 170 nM T67619 CGO6U5 54581103 IC50 = 690 nM T67619 CEKH90 54581104 IC50 = 9 nM T67619 C5LX1N 54581105 IC50 = 1100 nM T67619 CS76ZN 54581209 IC50 = 1000 nM T67619 CN4S9G 54581210 IC50 = 4400 nM T67619 CKD32N 54581211 IC50 = 6400 nM T67619 C7TQB1 54582142 IC50 = 310 nM T67619 CPS7O0 54582143 IC50 = 8 nM T67619 C8V9EK 54582198 IC50 = 1000 nM T67619 C3CHW4 54582239 IC50 = 26 nM T67619 CPT3M0 54582240 IC50 = 10 nM T67619 CI5G9H 54583166 IC50 = 3900 nM T67619 C43TQN 54583167 IC50 = 2100 nM T67619 CT0UG4 54583168 IC50 = 22800 nM T67619 CPBE35 54583205 IC50 = 300 nM T67619 C9X1PJ 54583206 IC50 = 180 nM T67619 CCO4G2 54584089 IC50 = 180 nM T67619 CFG10P 54584090 IC50 = 740 nM T67619 CXW98R 54584091 IC50 = 81 nM T67619 CA8QL7 54584179 IC50 > 20000 nM T67619 CBI49V 54585035 IC50 = 12 nM T67619 C2B3AQ 54585036 IC50 = 160 nM T67619 C3L9HR 54585126 IC50 = 500 nM T67619 C4AV1T 54586067 IC50 = 3400 nM T67619 CX63ZJ 54586068 IC50 = 4000 nM T67619 C87RCN 54586977 IC50 = 1200 nM T67619 CAWL73 54587085 IC50 > 20000 nM T67619 CB1G6U 54587086 IC50 = 6200 nM T67619 C1N2PW 54587087 IC50 = 1300 nM T67619 CE1ZK6 54759168 IC50 > 10000 nM T67619 C1XS2J 54760383 IC50 > 10000 nM T67619 C9ZFS1 54764923 IC50 > 100000 nM T67619 CPC5D2 56603995 IC50 = 10 nM T67619 CEBQ15 56604005 IC50 = 794 nM T67619 CFP56A 56604013 IC50 = 560 nM T67619 CM8JX1 56604907 IC50 = 10000 nM T67619 CN9QD7 56643097 IC50 > 10000 nM T67619 C0DGV4 56644346 IC50 = 528 nM T67619 C01BDZ 56644402 IC50 = 348 nM T67619 C65BKQ 56646651 IC50 = 387 nM T67619 C27YEM 56658554 IC50 = 70 nM T67619 C95GNR 56658555 IC50 = 40 nM T67619 CCV92H 56658556 IC50 = 250 nM T67619 CX25QL 56658684 IC50 = 110 nM T67619 C8G4SB 56662008 IC50 = 20 nM T67619 C49OIA 56662009 IC50 = 140 nM T67619 CAKY61 56662153 IC50 = 12650 nM T67619 CQGV57 56665612 IC50 = 30 nM T67619 C6U2OQ 56668926 IC50 = 2680 nM T67619 CH72SM 56669073 IC50 = 240 nM T67619 CC12UJ 56669074 IC50 = 2300 nM T67619 COB07T 56669075 IC50 = 7 nM T67619 C7M1CR 56672407 IC50 = 1510 nM T67619 C7Z4XQ 56672408 IC50 = 39 nM T67619 COJ3S1 56672409 IC50 = 140 nM T67619 CW23YA 56673235 IC50 = 920 nM T67619 C2C6IG 56673236 IC50 = 160 nM T67619 C50VCZ 56675790 IC50 = 3380 nM T67619 C4PNF2 56675791 IC50 = 1570 nM T67619 CT3B9L 56675792 IC50 = 120 nM T67619 C80YFG 56675793 IC50 = 350 nM T67619 CHSX82 56675794 IC50 = 20 nM T67619 CZMX67 56675913 IC50 = 2140 nM T67619 C3KEI5 56676565 IC50 = 590 nM T67619 C9KV5E 56679105 IC50 = 400 nM T67619 CIK9D5 56679106 IC50 = 80 nM T67619 CU9IT6 56679107 IC50 = 40 nM T67619 CSNQ62 56679108 IC50 = 6850 nM T67619 C5ZN6X 56682067 IC50 = 44 nM T67619 CWVS28 56682405 IC50 = 850 nM T67619 CI7T0B 56682406 IC50 = 200 nM T67619 CNVL06 56682407 IC50 = 190 nM T67619 CV7U9R 56682408 IC50 = 460 nM T67619 CBN3T6 56682409 IC50 = 330 nM T67619 C4OU6L 56682539 IC50 = 5800 nM T67619 CZX9O7 56682540 IC50 = 20440 nM T67619 CT4E8R 56832546 IC50 = 3600 nM T67619 C4Z0OC 56834890 Ki = 170 nM T67619 C67TJQ 56834891 Ki = 360 nM T67619 C32CID 56926598 Ki = 210 nM T67619 CV8Z5C 56926697 Ki = 230 nM T67619 CO43FQ 56926699 Ki = 10 nM T67619 C4GT2U 56926701 Ki = 100 nM T67619 CYN2F3 56953649 IC50 = 1042 nM T67619 CSP4N8 56954881 IC50 = 1262 nM T67619 C1DVM6 56955067 IC50 = 243 nM T67619 CSD5P3 56955068 IC50 = 926 nM T67619 CMZ9R5 56955069 IC50 = 199 nM T67619 CH49DB 56955070 IC50 = 8665 nM T67619 CV8LH9 56955071 IC50 = 787 nM T67619 CTZV87 56955180 IC50 = 8976 nM T67619 C3A1JB 56955181 IC50 = 301 nM T67619 CRK4A9 56955182 IC50 = 188 nM T67619 CIV4Y0 56955184 IC50 = 117 nM T67619 CQ31WL 56955185 IC50 = 193 nM T67619 C5NZQ7 56955186 IC50 = 465 nM T67619 CON3C4 56955187 IC50 = 2716 nM T67619 CK2T5P 56955280 IC50 = 1807 nM T67619 CO1QW7 56955281 IC50 = 5404 nM T67619 CR0ZC9 56955282 IC50 = 2668 nM T67619 C4HY7S 56955283 IC50 = 2135 nM T67619 CA3Y9U 56955284 IC50 = 2799 nM T67619 CP84GT 56955285 IC50 = 7024 nM T67619 C8EP9I 56955286 IC50 = 41722 nM T67619 CAK91L 56955954 IC50 > 3600 nM T67619 CS7U9L 56965952 IC50 = 5 nM T67619 C5USP1 57327769 IC50 = 830 nM T67619 CZYM98 57327842 IC50 = 800 nM T67619 CS49KB 57327913 IC50 = 880 nM T67619 CQ57PE 57345536 IC50 = 9026 nM T67619 CO0G4W 57391497 IC50 = 3100 nM T67619 CYC2K8 57394983 IC50 = 40200 nM T67619 CXC03J 57394984 IC50 = 16300 nM T67619 C8W6IG 57395117 IC50 > 30000 nM T67619 C0UDY9 57401151 IC50 > 30000 nM T67619 C3GD0Q 57403715 IC50 = 15000 nM T67619 CQP7E0 57750290 IC50 = 4 nM T67619 C1U3YR 57750299 IC50 = 3 nM T67619 CEY8W0 57750311 IC50 = 16 nM T67619 CNBO65 57750312 IC50 = 7 nM T67619 C2F9DS 57750315 IC50 = 30 nM T67619 CZ08KN 57750321 IC50 = 4 nM T67619 CUY8T6 57750329 IC50 = 149 nM T67619 CK4W1L 57750342 IC50 = 5 nM T67619 CM5X9L 57750343 IC50 = 276 nM T67619 C0TNP8 57750364 IC50 = 31 nM T67619 CBY5E4 57750369 IC50 = 5 nM T67619 CO6P5G 57750381 IC50 = 6 nM T67619 CSI9Y4 57750382 IC50 = 41 nM T67619 C6GH7X 57750391 IC50 = 31 nM T67619 CL7CW0 57750402 IC50 = 10 nM T67619 CA4G5W 57750407 IC50 = 4 nM T67619 CM7XL6 57750408 IC50 = 4 nM T67619 CY4Z8R 57750418 IC50 = 9 nM T67619 C8OY4I 57750420 IC50 = 42 nM T67619 CVK0G4 58056356 IC50 > 50000 nM T67619 C87LKR 58191080 IC50 = 75 nM T67619 CZPF92 58191081 IC50 = 6 nM T67619 CZA32V 58344912 IC50 = 1300 nM T67619 CL63DN 58344915 IC50 = 930 nM T67619 CPVF85 58344916 IC50 = 410 nM T67619 CD3LX9 58344922 IC50 = 16 nM T67619 CS8ZY7 58344924 IC50 = 51 nM T67619 C89NVR 58344941 IC50 = 110 nM T67619 COJ80E 58344944 IC50 = 1300 nM T67619 CU24IC 58344970 IC50 = 540 nM T67619 CYK74H 58344983 IC50 = 28 nM T67619 CRJ47B 58345005 IC50 = 3900 nM T67619 CIOV02 58345019 IC50 = 110 nM T67619 CY62SG 58345029 IC50 = 8 nM T67619 CTLW48 58345032 IC50 = 810 nM T67619 C6OX1S 58345043 IC50 = 14 nM T67619 CB6KU0 58345048 IC50 = 260 nM T67619 CM5HE1 58345070 IC50 < 12 nM T67619 CP23UB 58345084 IC50 = 740 nM T67619 C7VZE0 58345118 IC50 = 660 nM T67619 CO18NP 58345151 IC50 = 24 nM T67619 CN27OH 58345157 IC50 = 250 nM T67619 CNO51P 58345162 IC50 > 300000 nM T67619 CPT41Z 58345166 IC50 = 35 nM T67619 CV61YJ 58345169 IC50 = 33 nM T67619 CW6SC9 58345215 IC50 = 720 nM T67619 CFLZ87 58345232 IC50 = 15 nM T67619 CYBT41 58345302 IC50 = 95 nM T67619 CV3O1E 58345313 IC50 = 35 nM T67619 C4PE7X 58345314 IC50 = 49 nM T67619 C8X3WB 58458198 IC50 = 8548 nM T67619 C20XPF 58458267 IC50 > 2000 nM T67619 CP85TJ 58458278 IC50 = 2 nM T67619 CT79LH 58458379 IC50 = 81 nM T67619 C6BPR2 58985201 IC50 > 30000 nM T67619 CT3EW2 59292007 IC50 > 1000 nM T67619 CB3RU7 59446654 IC50 = 820 nM T67619 CXJ63M 59603829 IC50 > 100000 nM T67619 CQEU96 59603842 IC50 = 80 nM T67619 CPVD45 59670809 IC50 = 12 nM T67619 C32WHR 59670989 IC50 = 12 nM T67619 CDWQ04 59671004 IC50 = 18 nM T67619 C43HZT 59671085 IC50 = 68 nM T67619 C0BRA5 59671144 IC50 = 1454 nM T67619 CEYW16 59671148 IC50 = 5 nM T67619 C50NWX 59671151 IC50 = 3 nM T67619 CZH4W5 59671179 IC50 = 367 nM T67619 C8FY0G 59671180 IC50 = 3 nM T67619 CVRS14 59688971 IC50 = 8 nM T67619 COH62U 60097413 IC50 > 5000 nM T67619 C1MR8Q 60097495 IC50 > 10000 nM T67619 CTXU08 60102494 IC50 = 24660 nM T67619 C5O2NT 60155007 IC50 > 300000 nM T67619 CSK31U 60155091 IC50 = 58000 nM T67619 CIP61J 60155092 IC50 > 300000 nM T67619 CGF0Y3 60155093 IC50 = 5900 nM T67619 CD3KZ6 60155094 IC50 = 185000 nM T67619 C4U0PT 60155095 IC50 > 300000 nM T67619 CC3MB4 60155179 IC50 = 1700 nM T67619 C8YB4E 60155180 IC50 = 8800 nM T67619 C2TQK4 60155269 IC50 = 320 nM T67619 C9QB8G 60155270 IC50 = 270 nM T67619 CDTW29 60155456 IC50 = 13000 nM T67619 CM6NF2 60155627 IC50 = 36 nM T67619 C62SQG 60155628 IC50 = 13 nM T67619 COS39T 60155629 IC50 = 3.7 nM T67619 CSZA16 60155724 IC50 > 3600 nM T67619 C4SGZ6 60165992 IC50 > 100000 nM T67619 C98NOD 60165993 IC50 > 100000 nM T67619 C3WIX5 60165994 IC50 > 100000 nM T67619 C0G5WC 60165995 IC50 = 41000 nM T67619 CEQ07N 60166135 IC50 > 100000 nM T67619 CRV13A 60166136 IC50 > 100000 nM T67619 CLP62H 60166137 IC50 = 75000 nM T67619 C9X0ZC 60166139 IC50 > 100000 nM T67619 CWPZ07 60166141 IC50 > 100000 nM T67619 CK6WO0 66552478 IC50 < 10000 nM T67619 C1HSE0 67035086 IC50 = 7000 nM T67619 CUJ28O 67112053 IC50 = 4 nM T67619 C2ZJC1 67113434 IC50 = 2460 nM T67619 CZ3P5I 67160938 IC50 = 5 nM T67619 C5KOD3 67161433 IC50 = 9 nM T67619 CT04DK 67161469 IC50 = 6 nM T67619 CE5M9O 67161513 IC50 = 5 nM T67619 CG6XQ3 67161715 IC50 = 74 nM T67619 CP60OA 67161792 IC50 = 7 nM T67619 C1YX5L 67162199 IC50 = 1271 nM T67619 CNXU89 67162253 IC50 = 53 nM T67619 CPB2W6 67162323 IC50 = 3589 nM T67619 C2G7FT 67162514 IC50 = 13 nM T67619 CIY82C 67162897 IC50 = 56 nM T67619 CV63UL 67240318 IC50 > 10000 nM T67619 CP8OI2 67304551 IC50 = 270 nM T67619 CY76UR 67305743 IC50 = 2.7 nM T67619 C3UKG8 67312397 IC50 = 2.3 nM T67619 CM6TZ3 67312506 IC50 = 6 nM T67619 C8I7GC 68293638 IC50 > 10000 nM T67619 C5DGR9 69036886 IC50 = 10000 nM T67619 CS8UF1 70675988 IC50 = 3 nM T67619 C2W5BX 70675991 IC50 = 902 nM T67619 CUJA60 70676312 IC50 = 3 nM T67619 CRBW21 70676316 IC50 = 12 nM T67619 CGX49K 70676464 IC50 = 3 nM T67619 CQ82HN 70682337 IC50 = 1660 nM T67619 CPH18V 70683399 IC50 = 174 nM T67619 C4E7LN 70689727 IC50 = 240 nM T67619 CP6MQ7 70692884 IC50 = 810 nM T67619 CBE4Q7 70696974 IC50 = 5020 nM T67619 C1IEJ2 70789254 IC50 = 14000 nM T67619 C8T7ZP 70789255 IC50 = 1600 nM T67619 CH0B8N 70789756 IC50 > 30000 nM T67619 C91HPI 71300299 IC50 > 5000 nM T67619 CKT60L 71455860 Ki > 8000 nM T67619 CW8JR3 71510528 IC50 = 1730 nM T67619 C9DIK2 71512060 IC50 > 10000 nM T67619 CP05SQ 71526878 IC50 < 10 nM T67619 CCN01X 71547862 IC50 > 10000 nM T67619 CA3O6K 71552696 IC50 > 30000 nM T67619 C1NPL0 71552941 IC50 > 30000 nM T67619 CA4PS8 71552942 IC50 > 30000 nM T67619 C3UA9C 71553011 IC50 = 30000 nM T67619 CEZ15Y 71553012 IC50 = 18580 nM T67619 CVIA91 71553085 IC50 = 30000 nM T67619 C1TR3O 71553152 IC50 = 30000 nM T67619 CB3SO2 71567006 IC50 > 10000 nM T67619 CDJY72 71568837 IC50 > 10000 nM T67619 CBCW18 71571355 IC50 = 2070 nM T67619 CS37NG 71582865 IC50 = 5500 nM T67619 C7OZV5 71582867 IC50 = 6200 nM T67619 C6EOM7 71582869 IC50 = 5000 nM T67619 CP7AU3 71582871 IC50 = 3000 nM T67619 CCF67M 71582873 IC50 = 6900 nM T67619 C1NE2W 71582969 IC50 = 19100 nM T67619 CQV96E 71583048 IC50 = 1313 nM T67619 CSPR52 71583049 IC50 = 2753 nM T67619 CNT5F3 71583050 IC50 = 183 nM T67619 CH7I0W 71583051 IC50 = 1192 nM T67619 C1BG2L 71584579 IC50 = 3100 nM T67619 CQ0K5B 71584581 IC50 = 2000 nM T67619 CJBD60 71584583 IC50 = 10900 nM T67619 C4N7XQ 71584585 IC50 = 7000 nM T67619 C1GDL2 71602514 IC50 = 21.6 nM T67619 CHV4N8 71602515 IC50 = 5.24 nM T67619 C7YVU4 71602573 IC50 = 22 nM T67619 C90PSW 71602574 IC50 = 11.2 nM T67619 C34HNA 71602575 IC50 = 288 nM T67619 CM06KQ 71602576 IC50 = 23.8 nM T67619 CXSI14 71718330 IC50 > 100000 nM T67619 C1TM3P 71720141 IC50 > 100000 nM T67619 C0DL3F 72698602 IC50 = 2.16 nM T67619 CHM7O3 72946668 IC50 = 13670 nM T67619 C71GBE 73349501 IC50 = 1260 nM T67619 C3UC9H 73891099 IC50 = 2150 nM T67619 CV8QX0 76310169 IC50 > 30000 nM T67619 C3B8YH 76310394 IC50 = 470 nM T67619 CU0RT2 76310395 IC50 = 1430 nM T67619 C5BV3G 76310396 IC50 = 38 nM T67619 CLPF12 76311068 IC50 = 1830 nM T67619 CZAB97 76314060 IC50 = 1320 nM T67619 CYM1A9 76317612 IC50 = 160 nM T67619 C4J0OI 76317613 IC50 = 170 nM T67619 C8K6VZ 76317614 IC50 = 1250 nM T67619 C1OI4C 76317615 IC50 = 640 nM T67619 C1Y2HB 76318262 IC50 = 1830 nM T67619 C81EGJ 76318263 IC50 = 436.52 nM T67619 CL3VY9 76321344 IC50 = 220 nM T67619 CN6M7G 76321346 IC50 = 740 nM T67619 CA5L4W 76324771 IC50 > 30000 nM T67619 C6L9UI 76325588 IC50 = 4320 nM T67619 C9GO0P 76328313 IC50 = 23200 nM T67619 CYK65P 76328511 IC50 = 740 nM T67619 CRD20J 76332186 IC50 = 1260 nM T67619 C2IYA8 76332187 IC50 = 370 nM T67619 CP89GI 76332188 IC50 = 480 nM T67619 CI67WH 76332189 IC50 = 650 nM T67619 CHAP09 76332810 IC50 = 16.98 nM T67619 CJ2T9E 76332983 IC50 > 10000 nM T67619 C39FTZ 76335685 IC50 > 100000 nM T67619 CH2B4A 76335825 IC50 = 900 nM T67619 CN4CI1 76335826 IC50 = 1100 nM T67619 C6SQ4M 76336432 IC50 = 7.7 nM T67619 CPG3A5 86302574 IC50 > 30000 nM T67619 C1HW4B 89735655 IC50 = 870 nM T67619 CY0UC4 90645194 IC50 > 10000 nM T67619 CE72RT 90645487 IC50 = 200 nM T67619 CT1R6X 90645488 IC50 > 100000 nM T67619 CUR14N 90645489 IC50 = 4480 nM T67619 CUQ8M6 90645490 IC50 > 100000 nM T67619 C4U7KS 90645491 IC50 = 16130 nM T67619 C0SL1R 90645492 IC50 > 100000 nM T67619 CG71IS 90645493 IC50 = 4680 nM T67619 C1NR3K 90664901 IC50 = 5 nM T67619 CAU45T 91971978 IC50 > 15000 nM T67619 CLB50N 102300642 IC50 = 31330 nM T67619 CY6BK1 118408862 IC50 = 21.6 nM T67619 C4E2HN 118408899 IC50 = 72.3 nM T67619 CY7BI2 118706214 IC50 > 10000 nM T67619 C3KLI5 118723185 IC50 > 100000 nM T67619 CQCX41 118737057 IC50 > 10000 nM T67619 C31YGS 122189176 IC50 > 1000 nM T67619 CC48FJ 122189177 IC50 > 1000 nM T67619 CPGO14 126504238 IC50 = 2.9 nM T67619 C8WJF6 127027348 IC50 = 87600 nM T67619 C97SCV 127048164 IC50 = 1400 nM T67619 CYE59O 127049175 IC50 = 1480 nM T67619 CU4B1H 127049214 IC50 = 920 nM T67619 CJ5PL6 127049215 IC50 = 320 nM T67619 CTW06Y 127049216 IC50 = 360 nM T67619 C7WQ0S 127049217 IC50 = 71 nM T67619 CGI93L 127049218 IC50 = 920 nM T67619 CC0PL7 127049219 IC50 = 2020 nM T67619 CT5YD4 127049827 IC50 = 440 nM T67619 CAF85B 127052883 IC50 = 1260 nM T67619 CAY08K 127052885 IC50 = 850 nM T67619 CBJD38 127052886 IC50 = 1910 nM T67619 CTK5Y3 127052920 IC50 = 390 nM T67619 CO0U2R 127052921 IC50 = 61 nM T67619 C0FM1R 130196825 IC50 > 30000 nM T67619 CO47QJ 133054002 IC50 = 3 nM T67619 CT0GQ6 135197577 IC50 > 10000 nM T67619 C87VKA 135197594 IC50 > 10000 nM T67619 CQXS07 135197635 IC50 > 10000 nM T67619 C7KXF1 135197643 IC50 > 10000 nM T67619 C2KFH7 135398497 Ki > 2000 nM T67619 CU60YC 135431661 IC50 = 26890 nM T67619 CC4U9W 135443345 IC50 = 1.2 nM T67619 C9J4ES 135503073 IC50 = 62 nM T67619 CTJ48K 135524085 IC50 > 10000 nM T67619 CUT1W7 135524168 IC50 > 10000 nM T67619 CRJ45X 135589980 IC50 = 4430 nM T67619 CX4ZB3 135863110 IC50 = 10200 nM T67619 CYDM01 135891431 IC50 > 10000 nM T67619 CXM24U 135971437 IC50 = 15 nM T67619 C13AFE 135971438 IC50 = 500 nM T67619 CAH06E 135971439 IC50 = 10 nM T67619 C9SL8R 135971440 IC50 = 63 nM T67619 CCO83V 135971441 IC50 = 3 nM T67619 CHA4N2 136013680 IC50 > 10 nM T67619 CK94UW 136036657 IC50 = 34 nM T67619 CIYD68 136043776 IC50 = 6.5 nM T67619 CO16JK 136099766 IC50 = 71 nM T67619 C3ZS9L 136099767 IC50 = 127 nM T67619 CLB4O7 136099768 IC50 = 69 nM T67619 C6HW4E 136206295 IC50 > 100000 nM T67619 CU9P3M 136206296 IC50 > 100000 nM T67619 C1YUD0 136219394 IC50 > 10 nM T67619 CIU8W3 136254389 IC50 > 10 nM T67619 C5MZV6 137189918 IC50 = 1850 nM T67619 CMCD09 137189935 IC50 = 3230 nM T67619 C6MYZ0 137226336 IC50 = 7190 nM T67619 CT8EV4 137226337 IC50 = 8610 nM T67619 CC9S1D 137226351 IC50 = 16350 nM T67619 CI1E8V 137634241 IC50 > 10000 nM T67619 C8GQD5 137636872 IC50 = 608 nM T67619 CC73PA 138911338 IC50 = 1.37 nM T67619 CO6VM3 141404226 IC50 = 18 nM T67619 CMVP74 141404248 IC50 > 40 nM T67619 CC8UO6 141404250 IC50 = 2.9 nM T67619 CLC5X6 141404253 IC50 = 20.3 nM T67619 CTZI67 141404259 IC50 = 27.1 nM T67619 CP9GB3 141404261 IC50 = 7.6 nM T67619 C5ZMH7 141404263 IC50 = 35.6 nM T67619 CL2CA3 141404267 IC50 = 26.5 nM T67619 CA2WM4 141404269 IC50 > 40 nM T67619 C4SXV6 141404272 IC50 = 4.3 nM T67619 C6VB3O 145925651 IC50 >= 5000 nM T67619 CJK8E2 145949482 IC50 = 56 nM T67619 CYH7W1 145949795 IC50 = 482 nM T67619 CCY2L0 145949821 IC50 = 115 nM T67619 C5ZC7N 145951833 IC50 = 12 nM T67619 CK95RI 145954638 IC50 = 313 nM T67619 C1LNV7 145955342 IC50 = 1.72 nM T67619 CJWB07 145955381 IC50 = 98330 nM T67619 C0J9UP 145956191 IC50 = 138330 nM T67619 C6UYP8 145957119 IC50 = 176 nM T67619 CSXG01 145957159 IC50 = 311 nM T67619 C92EJD 145957936 IC50 = 980 nM T67619 CJF68H 145958278 IC50 = 27500 nM T67619 CQK7C4 145958439 IC50 = 640 nM T67619 CQ5L2P 145958887 IC50 = 8.2 nM T67619 C7SU8K 145959258 IC50 = 4.7 nM T67619 CQYX04 145959319 IC50 = 432 nM T67619 CFOG23 145960003 IC50 = 251 nM T67619 C65YWX 145964882 IC50 > 10000 nM T67619 CHC3T0 145965031 IC50 > 10000 nM T67619 CP92ZF 145965329 IC50 > 10000 nM T67619 C9HXI4 145966620 IC50 > 10000 nM T67619 CQE9M5 145966810 IC50 > 10000 nM T67619 C1EH6C 145967078 IC50 > 10000 nM T67619 CDNC31 145967951 IC50 > 500 nM T67619 CWJ12M 145969155 IC50 > 10000 nM T67619 CGW5S1 145969844 IC50 > 10000 nM T67619 CB8R3A 145970271 IC50 > 10000 nM T67619 CWTM19 145971215 IC50 = 738 nM T67619 C40VIL 145972979 IC50 > 10000 nM T67619 CO39BH 145973343 IC50 = 5.6 nM T67619 CJP7A0 145973531 IC50 = 14.1 nM T67619 CQBY19 145974023 IC50 = 1900 nM T67619 C4OMF0 145976589 IC50 = 1.9 nM T67619 C4X7CT 145977420 IC50 > 10000 nM T67619 CLA57T 145978300 IC50 > 10000 nM T67619 CJM2O4 145978607 IC50 = 1.5 nM T67619 CV9L5H 145978676 IC50 = 1.8 nM T67619 C41TSL 145980453 IC50 = 32.9 nM T67619 CZ34CG 145981520 IC50 = 26.9 nM T67619 CSXW63 145988300 IC50 = 51.9 nM T67619 CX1JI9 145989967 IC50 = 30.5 nM T67619 CA1T2G 145990354 IC50 = 66.6 nM T67619 CNR64J 145991965 IC50 = 24.3 nM T67619 CSU93V 155077019 IC50 = 0.98 nM T67619 C47WVH 155510889 IC50 = 529.5 nM T67619 CT56FP 155511113 IC50 = 1 nM T67619 C4XJ3M 155511115 IC50 = 127.4 nM T67619 CQX1T3 155512930 IC50 = 10.2 nM T67619 CE6X7Y 155513578 IC50 = 3.24 nM T67619 CU0Y4W 155513852 IC50 = 29.8 nM T67619 CH02UG 155514203 IC50 < 10000 nM T67619 CC5G1K 155514612 IC50 = 27.3 nM T67619 CB21RJ 155515141 IC50 = 3.29 nM T67619 C9BT0N 155515321 IC50 = 13.7 nM T67619 C2BPO4 155515456 IC50 = 181.8 nM T67619 CQV81J 155516726 IC50 = 17.3 nM T67619 C0JS3R 155517116 IC50 = 5.46 nM T67619 CG1A3H 155517747 IC50 = 57.7 nM T67619 CH2S3X 155517930 IC50 = 73.5 nM T67619 CQX0D7 155518023 IC50 = 10.6 nM T67619 C2P0DV 155518372 IC50 = 709.6 nM T67619 C5ICP0 155518486 IC50 = 149.3 nM T67619 CFL74D 155519231 IC50 = 7.98 nM T67619 C1DF7C 155519583 IC50 = 1.94 nM T67619 C2EP0N 155520797 IC50 = 12.41 nM T67619 CMDO31 155520865 IC50 = 3646 nM T67619 CXM73F 155521242 IC50 = 13.7 nM T67619 CE9IK1 155521336 IC50 = 8.78 nM T67619 CG69OE 155521843 IC50 = 2.56 nM T67619 C1PC3M 155521934 IC50 = 1.26 nM T67619 C6WAB4 155521997 IC50 = 215 nM T67619 C60CES 155523241 IC50 = 321.6 nM T67619 C4LKN7 155523722 IC50 > 1000 nM T67619 C12XTS 155523979 IC50 = 1.8 nM T67619 C89GPZ 155525215 IC50 = 62.2 nM T67619 CL5DR0 155525783 IC50 = 3 nM T67619 CLQ50N 155525830 IC50 = 211.9 nM T67619 CXD6N9 155528054 IC50 = 65.2 nM T67619 C9XKJ3 155528122 IC50 = 2.49 nM T67619 C47TOX 155528238 IC50 = 101 nM T67619 CETK89 155528489 IC50 = 538 nM T67619 C39PEC 155529638 IC50 < 10000 nM T67619 COKA05 155531035 IC50 < 10000 nM T67619 C86MSV 155531147 IC50 = 6.4 nM T67619 CSE1M5 155531643 IC50 = 35.6 nM T67619 CE4LB3 155532531 IC50 = 10.44 nM T67619 CWU2L1 155532647 IC50 = 46.9 nM T67619 C47KDV 155534523 IC50 = 3.79 nM T67619 C15BDE 155534728 IC50 = 104.1 nM T67619 CLN3G8 155535243 IC50 = 17.6 nM T67619 CNA5M9 155536532 IC50 = 1566 nM T67619 CYKO64 155537875 IC50 = 2.64 nM T67619 CWN30S 155538720 IC50 = 5.65 nM T67619 CAO50V 155539664 IC50 = 101.6 nM T67619 C1MW0T 155540708 IC50 < 10000 nM T67619 C9LXF1 155541357 IC50 = 29.4 nM T67619 CUQ0I5 155541401 IC50 = 2.74 nM T67619 C91ARO 155541435 IC50 = 5.99 nM T67619 CF3B6R 155542062 IC50 = 4.47 nM T67619 C9ITP8 155543671 IC50 = 230.2 nM T67619 CS9MO6 155543688 IC50 = 76.6 nM T67619 C6NB5M 155543985 IC50 = 70.4 nM T67619 C62BHG 155544807 IC50 = 3.31 nM T67619 CP83YC 155545670 IC50 = 5.1 nM T67619 C79FLK 155545798 IC50 = 187.9 nM T67619 CJNL79 155546504 IC50 = 3.4 nM T67619 CV7T6F 155546619 IC50 > 1000 nM T67619 CLU14D 155547124 IC50 = 51.2 nM T67619 CI93AE 155548647 IC50 = 7.2 nM T67619 CE9UZ8 155549694 IC50 = 50.3 nM T67619 C26IZH 155552261 IC50 = 6.41 nM T67619 CH4UX7 155552337 IC50 = 448.9 nM T67619 C70ELS 155552548 IC50 > 1000 nM T67619 C5AH8Y 155552974 IC50 = 162.5 nM T67619 C8GA9Q 155553579 IC50 = 35.3 nM T67619 CS12YQ 155553782 IC50 = 99.9 nM T67619 CHS21A 155553831 IC50 = 17 nM T67619 CBZF15 155555139 IC50 < 10000 nM T67619 CX90VQ 155555430 IC50 < 10000 nM T67619 C2PI8G 155556173 IC50 = 48.9 nM T67619 C13SAT 155556233 IC50 = 1.41 nM T67619 CV3GE1 155556291 IC50 = 17.3 nM T67619 CNB0P5 155556393 IC50 = 2.5 nM T67619 CDL0Q9 155558294 IC50 = 199.1 nM T67619 CJGI53 155559701 IC50 = 269.8 nM T67619 C97KIE 155560308 IC50 = 7.01 nM T67619 CUN71C 155560648 IC50 = 500 nM T67619 C5R2QD 155561801 IC50 = 8 nM T67619 CS73HF 155562030 IC50 = 222.2 nM T67619 CGJ67F 155562297 IC50 > 1000 nM T67619 C04OXM 155562654 IC50 < 10000 nM T67619 CY48VH 155562963 IC50 = 191 nM T67619 CG95WV 155563831 IC50 = 1.9 nM T67619 C3ZVW9 155565280 IC50 = 9 nM T67619 CZ5R2M 155565595 IC50 = 31.2 nM T67619 C6Q0NX 155566205 IC50 = 40 nM T67619 CEIW13 155566807 IC50 = 72 nM T67619 CW2Z7R 155567578 IC50 = 255.3 nM T67619 CM10TL 155568505 IC50 = 3.4 nM T67619 CKM67J 155568657 IC50 = 3.95 nM T67619 C14GTU 155568758 IC50 = 9.3 nM T67619 CS81XG 155569192 IC50 = 3.13 nM T67619 D00ATA 5908088 IC50 = 2300 nM T67619 D00ERW 44444843 Ki = 3698 nM T67619 D00HVA 11624601 Ki > 8200 nM T67619 D03DZO 11715767 IC50 > 10000 nM T67619 D04PEI 11467730 IC50 > 50000 nM T67619 D04ZWF 53396311 IC50 > 5000 nM T67619 D05APZ 135398501 IC50 = 58 nM T67619 D06HVH 54613583 IC50 > 10000 nM T67619 D06QWO 14824655 IC50 > 10 ug.mL-1 T67619 D07OXC 11650194 IC50 > 100000 nM T67619 D08HFG 24809764 IC50 > 10000 nM T67619 D09FFE 449241 IC50 = 1600 nM T67619 D09HVH 135566652 IC50 > 10 nM T67619 D09XIL 11396738 IC50 > 125000 nM T67619 D0A1CM 5281855 IC50 = 3340 nM T67619 D0AY0F 70698427 IC50 > 10000 nM T67619 D0CM6T 11314340 Ki = 11 nM T67619 D0D9PD 11656591 IC50 > 5000 nM T67619 D0DQ6Z 8530 IC50 = 10980 nM T67619 D0EU1R 46215815 IC50 > 10000 nM T67619 D0F0AU 44405988 IC50 > 20000 nM T67619 D0F8HX 12967404 IC50 = 149 nM T67619 D0G3SZ 6918469 IC50 > 10 ug.mL-1 T67619 D0GD8Y 3006531 IC50 = 60000 nM T67619 D0I1FJ 11393719 IC50 = 200 nM T67619 D0L2WP 46225540 IC50 = 1 nM T67619 D0M9QJ 44240850 IC50 = 6300 nM T67619 D0ME9B 46868971 IC50 > 10 nM T67619 D0O6OH 71553154 IC50 = 3100 nM T67619 D0OX1T 10172943 Ki = 0.16 nM T67619 D0Q3KS 9957049 IC50 > 10000 nM T67619 D0Q3NG 11715520 Ki > 8200 nM T67619 D0RZ1H 11424128 IC50 = 19700 nM T67619 D0S7IE 11658882 Ki > 8200 nM T67619 D0T8NU 16757525 IC50 > 4000 nM T67619 D0UN9O 3385203 IC50 >= 10000 nM T20973 D0EG1I 9926791 IC50 > 10000 nM T20973 D00UZR 5330286 IC50 > 10000 nM T20973 D05ADP 160355 IC50 = 270 nM T20973 D0LF1U 5287969 IC50 = 170 nM T20973 D0P0KN 16739650 IC50 = 3 nM T20973 D0PL7P 24983461 IC50 = 23 nM T20973 D0A3MV 448014 IC50 = 100000 nM T20973 D00BPA 4592 IC50 = 3000 nM T20973 D0D3PX 46926350 IC50 = 1 nM T20973 CHR3Z9 5097 IC50 = 160 nM T20973 C1ZG2U 449087 IC50 = 114 nM T20973 CZU0A4 5479542 IC50 > 10000 nM T20973 C8O4ZA 6538904 IC50 > 100000 nM T20973 C1KHR3 6538905 IC50 = 40000 nM T20973 C0VLD2 6538906 IC50 = 14000 nM T20973 C36NRA 6538907 IC50 = 13000 nM T20973 C34REF 6538908 IC50 > 100000 nM T20973 COS29U 6538909 IC50 > 100000 nM T20973 C50PWH 6538910 IC50 > 100000 nM T20973 CU17AZ 6538911 IC50 > 100000 nM T20973 CMV28P 6538912 IC50 > 100000 nM T20973 C7ZBQ5 6538913 IC50 > 100000 nM T20973 CNR9G3 6538914 IC50 = 2400 nM T20973 CZ36MO 6538915 IC50 = 1300 nM T20973 C6IV4B 6538916 IC50 = 8000 nM T20973 CXU3H2 6538917 IC50 = 2300 nM T20973 CE1QL2 6538918 IC50 = 2300 nM T20973 C6F5WG 6538919 IC50 = 3500 nM T20973 CL4Z8I 6538920 IC50 = 6000 nM T20973 C7DT1S 6538921 IC50 = 2000 nM T20973 CGH45F 6538922 IC50 = 1300 nM T20973 CJGK38 6538923 IC50 = 400 nM T20973 CMN3A9 6538924 IC50 = 700 nM T20973 CXC4R3 6538925 IC50 = 35000 nM T20973 C5K8QG 6538926 IC50 = 160 nM T20973 CNDE01 6538927 IC50 = 2400 nM T20973 C4VZ3Y 6538928 IC50 = 13000 nM T20973 C5N3IH 6538929 IC50 = 500 nM T20973 CID0S2 6538930 IC50 > 100000 nM T20973 C7JC5M 6538932 IC50 = 400 nM T20973 C1LI8N 6538935 IC50 = 340 nM T20973 CUFR51 6538960 IC50 = 500 nM T20973 C5KW8Q 6538961 IC50 = 230 nM T20973 C6IWQ1 6538962 IC50 = 300 nM T20973 C0RCH9 6538963 IC50 = 600 nM T20973 CX2TI8 6538964 IC50 = 260 nM T20973 CXV4N7 6538965 IC50 = 300 nM T20973 CYCI38 6538966 IC50 = 300 nM T20973 C13IWP 6538967 IC50 = 400 nM T20973 CAO4T9 6538968 IC50 = 500 nM T20973 C1NY5R 6538969 IC50 = 500 nM T20973 CS20UD 7311753 IC50 < 50000000 nM T20973 CQ4PX0 9815202 IC50 = 16 nM T20973 CLW4V7 9835236 IC50 = 183 nM T20973 CH4M1G 9836448 IC50 = 190 nM T20973 CHO8J3 9858435 IC50 = 44 nM T20973 C2QVB5 9879866 IC50 = 41 nM T20973 CJ30OC 9881657 IC50 = 102 nM T20973 CLP53M 9901306 IC50 = 48 nM T20973 CFQZ60 9901793 IC50 = 8 nM T20973 C5WR3M 9921612 IC50 = 25 nM T20973 CK81XG 9923299 IC50 = 44 nM T20973 CI8HJ7 9923300 IC50 = 5 nM T20973 CTLS37 9967013 IC50 = 10 nM T20973 CM9NI0 9967051 IC50 = 13 nM T20973 C52YXF 10132219 IC50 = 12 nM T20973 C7PU4Z 10224714 IC50 = 225 nM T20973 CIU4R3 10268127 IC50 = 13 nM T20973 CA9T8Q 10291035 IC50 = 13 nM T20973 C5X4NT 10308461 IC50 = 54 nM T20973 C2B0IU 10421236 IC50 = 3500 nM T20973 C37ASK 10449986 IC50 = 131 nM T20973 C04NLR 11245667 IC50 > 50000 nM T20973 CMZ6Q7 11277469 IC50 = 30000 nM T20973 CUM15V 11358339 IC50 > 50000 nM T20973 C8KPE4 11380176 IC50 > 50000 nM T20973 C4PSB5 11437879 IC50 > 50000 nM T20973 CTG83F 11539329 Ki > 9300 nM T20973 CMIL86 11590363 Ki > 9300 nM T20973 C9T6SC 11640926 Ki > 9300 nM T20973 CVC2S4 11722798 IC50 = 79 nM T20973 CP7AH3 11755812 IC50 = 50000 nM T20973 CHR92S 11858109 IC50 > 100000 nM T20973 CFPW41 16007116 Ki > 9300 nM T20973 C7BS2R 16037674 IC50 > 10000 nM T20973 CB2H4D 16037675 IC50 = 3000 nM T20973 CKR57M 16086104 IC50 > 25000 nM T20973 C16NRY 16086114 IC50 > 25000 nM T20973 CQG45C 16109001 IC50 = 100000 nM T20973 C1U8XW 16109036 IC50 > 100000 nM T20973 CGC34R 16118737 IC50 > 25000 nM T20973 C4V9QD 16760027 IC50 = 64 nM T20973 CIJ9X7 22170542 IC50 = 900 nM T20973 C8RWK9 22170582 IC50 = 4580 nM T20973 C36FIU 22170855 IC50 = 1150 nM T20973 C5WJB7 22731378 IC50 = 3990 nM T20973 CSE84O 22731387 IC50 = 7 nM T20973 CNYQ64 23074669 IC50 > 100000 nM T20973 CFMQ08 24370907 IC50 > 100000 nM T20973 C4Z9CN 24769780 IC50 > 100000 nM T20973 CT4RG0 24800068 IC50 = 5900 nM T20973 CZ48LS 24825971 IC50 = 25000 nM T20973 CK4RG2 25167767 IC50 = 4329 nM T20973 CD6Y0G 25268197 IC50 > 50000 nM T20973 CR59TN 25268198 IC50 > 50000 nM T20973 C1DR5Z 25268199 IC50 > 50000 nM T20973 CV4N5C 25268555 IC50 > 50000 nM T20973 CPM85N 25268556 IC50 > 50000 nM T20973 CT7EB2 25268557 IC50 > 50000 nM T20973 CWB2K9 25268558 IC50 > 50000 nM T20973 C81HUL 25268559 IC50 > 50000 nM T20973 CU9E4P 42629114 IC50 > 10000 nM T20973 C5PIG4 44353568 IC50 = 340 nM T20973 CEX13C 44395851 IC50 = 3270 nM T20973 CH23AG 44395852 IC50 = 1570 nM T20973 CRYQ73 44395922 IC50 = 7670 nM T20973 C56KVN 44395923 IC50 = 91 nM T20973 C06KDB 44396065 IC50 = 621 nM T20973 CEFX64 44396098 IC50 = 1600 nM T20973 CI3Z6V 44396116 IC50 = 321 nM T20973 C3EUC7 44396151 IC50 = 390 nM T20973 CDGY20 44396152 IC50 = 6530 nM T20973 C4KGN0 44396173 IC50 = 64 nM T20973 C5HZF2 44413509 IC50 = 34 nM T20973 C3D4FG 44413527 IC50 > 10000 nM T20973 C3VRO9 44557921 IC50 > 10000 nM T20973 C6E2SC 45482700 IC50 > 10000 nM T20973 CZXH74 45482750 IC50 > 10000 nM T20973 C29PHE 46882055 IC50 = 80 nM T20973 CYBR24 46882056 IC50 = 11000 nM T20973 C2O8RZ 46886323 IC50 > 1000 nM T20973 C60GAV 46929544 IC50 > 8000 nM T20973 CP34VL 46929748 IC50 > 1000 nM T20973 CJ2E9Q 46929857 IC50 > 25000 nM T20973 CCL3R5 49867929 IC50 = 3000 nM T20973 CO1TP3 52947886 IC50 = 5 nM T20973 CH2O0D 52948241 IC50 = 25000 nM T20973 C2G3AY 54726684 IC50 > 25000 nM T20973 C1MR8Q 60097495 IC50 > 10000 nM T20973 CL1HY5 71212233 IC50 > 100000 nM T20973 CKX52R 71212291 IC50 > 100000 nM T20973 C0T2VB 71212317 IC50 > 100000 nM T20973 C5B8NS 71212337 IC50 > 100000 nM T20973 CSN04E 71212395 IC50 > 100000 nM T20973 C1OCW0 71212403 IC50 > 100000 nM T20973 CBX2I4 71212419 IC50 > 100000 nM T20973 CLS4R3 71212434 IC50 > 100000 nM T20973 CTF8M7 71212446 IC50 > 100000 nM T20973 C2Z8CX 71212514 IC50 > 100000 nM T20973 CBT7L3 71212517 IC50 > 100000 nM T20973 CKT60L 71455860 Ki = 416 nM T20973 CHY91V 71578307 IC50 > 100000 nM T20973 C0W2KX 71578373 IC50 > 100000 nM T20973 C6TX9R 71578374 IC50 > 100000 nM T20973 C2D1RN 71578375 IC50 > 100000 nM T20973 C73MEW 71578445 IC50 > 100000 nM T20973 C5NH3V 71578446 IC50 > 100000 nM T20973 CC65WU 71578447 IC50 > 100000 nM T20973 CIP6Q2 71578520 IC50 > 100000 nM T20973 CPJ19D 71578658 IC50 > 100000 nM T20973 C5W0GC 71578744 IC50 > 100000 nM T20973 CLZ59B 71578745 IC50 > 100000 nM T20973 CYG95S 72707651 IC50 = 1502 nM T20973 CNP0V5 72707724 IC50 = 1420 nM T20973 CU4A5Q 72707728 IC50 = 1356 nM T20973 CZAM98 72707790 IC50 = 1178 nM T20973 CP13FK 72707853 IC50 = 1093 nM T20973 CWR57U 78357763 IC50 = 222 nM T20973 C8D3XO 86765295 IC50 > 10000 nM T20973 C0GYK1 86765296 IC50 = 9000 nM T20973 CUY63S 90645193 IC50 > 10000 nM T20973 C26BSU 90666124 IC50 > 10000 nM T20973 CVQ1O6 90666126 IC50 > 10000 nM T20973 C5AN9J 90666128 IC50 > 10000 nM T20973 CP76NE 90666130 IC50 > 10000 nM T20973 C85GHD 90666131 IC50 > 10000 nM T20973 CRP9I5 90666132 IC50 > 10000 nM T20973 CWE9I2 91664021 IC50 > 10000 nM T20973 CW58AE 91664022 IC50 > 10000 nM T20973 CB25UZ 91664023 IC50 > 10000 nM T20973 C8W9KV 91844733 IC50 = 9400 nM T20973 CL64EZ 102287891 IC50 > 10000 nM T20973 C2NQ4S 102287892 IC50 > 10000 nM T20973 C8GB4Q 122181008 IC50 > 10000 nM T20973 CBQ94Z 122181009 IC50 > 10000 nM T20973 CT8CP2 122181010 IC50 > 10000 nM T20973 CB6IZ0 122181011 IC50 > 10000 nM T20973 C65BOF 122181012 IC50 > 10000 nM T20973 CO83PN 122181013 IC50 = 10000 nM T20973 C69ULZ 122181014 IC50 > 100000 nM T20973 CN14DV 122181015 IC50 > 10000 nM T20973 CIG8Y1 122181016 IC50 > 10000 nM T20973 CRJS41 122181017 IC50 > 10000 nM T20973 CVB03H 122181018 IC50 > 10000 nM T20973 C6SJ3X 122181019 IC50 > 10000 nM T20973 C8IM5O 122181020 IC50 > 10000 nM T20973 C7L5PG 122181021 IC50 > 10000 nM T20973 C58CJI 122181022 IC50 > 10000 nM T20973 CG2Z8B 122181023 IC50 > 10000 nM T20973 CC2G8N 122181024 IC50 > 10000 nM T20973 CM2DU7 122181025 IC50 > 10000 nM T20973 C5YB3O 122181096 IC50 > 10000 nM T20973 CV5BQ9 122181097 IC50 > 10000 nM T20973 CE2D6Q 122688235 IC50 = 183 nM T20973 CGL61V 122696308 IC50 = 165 nM T20973 CE6FA8 127029858 IC50 = 17 nM T20973 C5KAL0 127029899 IC50 = 8 nM T20973 C3TPV9 127029900 IC50 = 44 nM T20973 CL0MX6 127030495 IC50 = 2136 nM T20973 CS26ZM 127030546 IC50 = 229 nM T20973 C5L6BD 127030848 IC50 = 49 nM T20973 C1SP3H 127030849 IC50 = 5 nM T20973 CXCT36 127030850 IC50 = 1 nM T20973 C5Z7FV 127030851 IC50 = 9 nM T20973 CKZ97R 127032672 IC50 = 3600 nM T20973 CM56SN 127033880 IC50 = 179 nM T20973 C20SZO 127033881 IC50 = 422 nM T20973 CV28XG 127033882 IC50 = 4415 nM T20973 CIQ5W3 127034385 IC50 = 119 nM T20973 CJK4T6 127034420 IC50 = 21 nM T20973 CB2ZW7 127034421 IC50 = 5 nM T20973 CNA05R 127034422 IC50 = 114 nM T20973 CNH46J 127034423 IC50 = 37 nM T20973 CJ3M5I 134137436 Ki > 1000 nM T20973 C4OWM1 135403014 IC50 = 5 nM T20973 C9QI4V 135423788 IC50 > 10000 nM T20973 CEVL69 135423792 IC50 > 10000 nM T20973 CTAC32 135423796 IC50 > 10000 nM T20973 CJ2F7R 136238979 IC50 > 10000 nM T20973 CT3KB7 136238980 IC50 > 10000 nM T20973 C8JGC6 136238981 IC50 > 10000 nM T20973 CJDO36 136238982 IC50 > 10000 nM T20973 CY6M7W 136239000 IC50 > 10000 nM T20973 CF1V6K 136239001 IC50 > 10000 nM T20973 C8G7OB 136239002 IC50 > 10000 nM T20973 CH17EC 136239003 IC50 > 10000 nM T20973 C3IV7E 136239004 IC50 > 10000 nM T20973 C0PQ5H 136239005 IC50 > 10000 nM T20973 CZ76FY 136239019 IC50 > 10000 nM T20973 C4OQ1U 136240234 IC50 < 50000000 nM T20973 CFUZ87 136240995 IC50 = 3400 nM T20973 CO17AY 136252249 IC50 > 10000 nM T20973 CRB3M4 136609929 IC50 > 10000 nM T20973 C0A9VE 136609930 IC50 > 10000 nM T20973 CW5YL0 136609931 IC50 > 10000 nM T20973 C3DNL6 137349544 IC50 = 9000 nM T20973 CGK3Q6 137634367 IC50 = 4400 nM T20973 C4DRX1 137643187 IC50 = 8840 nM T20973 CA5N2M 137654694 IC50 = 3300 nM T20973 CS02AJ 137661113 IC50 = 81000 nM T20973 CB2J4N 145989210 IC50 = 1 nM T20973 CR2GW6 145994117 IC50 = 680 nM T20973 CLXN40 155565350 IC50 = 232 nM T20973 C8AOM4 11724428 IC50 = 6000 nM T20973 D00ERW 44444843 Ki > 9275 nM T20973 D00HVA 11624601 Ki > 9300 nM T20973 D01MNK 25125014 IC50 = 30 nM T20973 D03DZO 11715767 IC50 = 460 nM T20973 D04NGS 5330790 IC50 = 12.59 nM T20973 D07OXC 11650194 IC50 > 100000 nM T20973 D0F0AX 135413546 IC50 = 30 nM T20973 D0GN5Z 5281295 IC50 = 1500 nM T20973 D0H3EV 5005498 IC50 = 40 nM T20973 D0L3FK 5289419 IC50 = 65 nM T20973 D0OZ2S 11785878 IC50 > 10000 nM T20973 D0Q3NG 11715520 Ki > 9300 nM T20973 D0R1FT 4564 IC50 = 97000 nM T20973 D0S7IE 11658882 Ki > 9300 nM T20973 D0Y5RO 4566 IC50 = 480 nM T26983 C19ZQH 8699243 IC50 = 13000 nM T26983 C3NE8O 46931242 IC50 > 10000 nM T26983 C2P7SD 56577044 IC50 > 10000 nM T26983 CXY3E4 57720618 IC50 > 30000 nM T26983 C0WX5O 70679311 IC50 > 30000 nM T26983 CEW3R6 71598546 IC50 = 14500 nM T26983 CUD65X 73333125 IC50 > 10000 nM T26983 CHQ18I 73333126 IC50 > 10000 nM T26983 C9UDN1 73333127 IC50 > 10000 nM T26983 C9K1NV 73333128 IC50 = 8700 nM T26983 C4UE6G 73333129 IC50 > 10000 nM T26983 CV2SJ4 73333225 IC50 > 10000 nM T26983 CF8HO3 73333226 IC50 > 10000 nM T26983 CVH9F0 73333227 IC50 > 10000 nM T26983 C4PYG2 73333229 IC50 = 3500 nM T26983 CBJC52 73333322 IC50 > 10000 nM T26983 CVEN67 73334066 IC50 > 10000 nM T26983 CYL3M7 73334067 IC50 > 10000 nM T26983 C6T7YX 73334068 IC50 = 4700 nM T26983 C70XCT 73334069 IC50 = 7900 nM T26983 C8QWP1 73334070 IC50 > 10000 nM T26983 CR98DL 73334157 IC50 = 7400 nM T26983 CJD9C1 73334158 IC50 > 10000 nM T26983 CLRM71 73334159 IC50 > 10000 nM T26983 C43NER 73334160 IC50 > 10000 nM T26983 CD2HX4 73334161 IC50 > 10000 nM T26983 CC89FN 73334162 IC50 > 10000 nM T26983 COV3R1 73334262 IC50 > 10000 nM T26983 CZD0N1 73334263 IC50 > 10000 nM T26983 CU3KG0 73334264 IC50 > 10000 nM T26983 CMLV27 73334265 IC50 > 10000 nM T26983 CD0VK7 73334266 IC50 > 10000 nM T26983 C1SGJ3 73334267 IC50 > 10000 nM T26983 C3PYF5 73334361 IC50 > 10000 nM T26983 C8H9JF 73334363 IC50 > 10000 nM T26983 C8XE1J 73334364 IC50 > 10000 nM T26983 CN40ZI 73334365 IC50 > 10000 nM T26983 CF9GA5 73334366 IC50 > 10000 nM T26983 C69WLM 73334479 IC50 > 10000 nM T26983 CG32QB 73334480 IC50 > 10000 nM T26983 CVE0S2 73334481 IC50 > 10000 nM T26983 C2S8XN 73334482 IC50 > 10000 nM T26983 CXJP87 73334483 IC50 > 10000 nM T26983 C57KSE 73334484 IC50 > 10000 nM T26983 CAQ18T 73334592 IC50 > 10000 nM T26983 CA67YG 73334593 IC50 > 10000 nM T26983 CNS84D 73334594 IC50 > 10000 nM T26983 C93HWE 73334595 IC50 > 10000 nM T26983 C87UBE 73334596 IC50 > 10000 nM T26983 CKSY83 73334696 IC50 > 10000 nM T26983 C36QHM 73334697 IC50 > 10000 nM T26983 CF63HU 73334698 IC50 > 10000 nM T26983 CQBX27 73334699 IC50 > 10000 nM T26983 C0OW1V 73334700 IC50 = 10700 nM T26983 CG80NF 73349257 IC50 > 10000 nM T26983 COY1J2 73349259 IC50 > 10000 nM T26983 CNO9Z5 73350843 IC50 > 10000 nM T26983 C8U0ZX 73352326 IC50 > 10000 nM T26983 C2OXQ5 76314887 IC50 > 30000 nM T26983 C3X7EW 76314888 IC50 > 30000 nM T26983 C1YKN5 76314889 IC50 > 30000 nM T26983 C4E1BN 76318504 IC50 > 30000 nM T26983 CF76CT 76318505 IC50 = 21000 nM T26983 CLVA91 76318506 IC50 > 30000 nM T26983 C9LNK4 76318507 IC50 > 30000 nM T26983 CL87KC 76318508 IC50 > 30000 nM T26983 CET23F 76318509 IC50 > 30000 nM T26983 C01JLF 76322168 IC50 > 30000 nM T26983 C2SEM0 76322169 IC50 > 30000 nM T26983 CRH48X 76322170 IC50 > 30000 nM T26983 C5CZV2 76325789 IC50 > 30000 nM T26983 CS6GL0 76333019 IC50 > 30000 nM T26983 C7IUX5 76333020 IC50 > 30000 nM T26983 CZC8W2 76336632 IC50 > 30000 nM T26983 CYQ0B9 76336633 IC50 = 19400 nM T26983 CK2N0L 76336634 IC50 > 30000 nM T26983 CS4W5I 76336635 IC50 > 30000 nM T26983 CM6H9O 76336636 IC50 = 18400 nM T26983 CI1WN4 78673861 IC50 = 30000 nM T26983 C23NAI 91970648 IC50 = 14000 nM T26983 CM7Q6B 91970649 IC50 = 22000 nM T26983 D0W9RR 57339144 IC50 = 13700 nM T89592 D03VOJ 8768 IC50 = 239000 nM T89592 C54JUR 25043 IC50 = 141000 nM T89592 C70HVL 77888 IC50 = 137000 nM T89592 CPI2E4 80447 IC50 = 71600 nM T89592 C07AKH 786691 IC50 = 20000 nM T89592 CY4MC6 3505109 IC50 = 145000 nM T89592 CGN9J7 44267478 IC50 = 25000 nM T89592 CH4Q6A 145964401 IC50 = 6100 nM T89592 CHU61S 145964420 IC50 = 600 nM T89592 C6YCA8 145964710 IC50 = 700 nM T89592 CV6F7L 145966788 IC50 = 600 nM T89592 CBWX17 145967285 IC50 = 900 nM T89592 COR9X3 145972736 IC50 = 700 nM T89592 CQ0M2X 145972809 IC50 = 7500 nM T89592 CF95RZ 145972878 IC50 = 600 nM T89592 CXI0D1 145975081 IC50 = 700 nM T89592 CG84ZR 145975487 IC50 = 400 nM T89592 C91FOT 145976006 IC50 = 800 nM T89592 C3F4UH 145978039 IC50 = 500 nM T11615 D02ZTJ 5339 IC50 = 160 nM T11615 D0C4YC 4075 IC50 > 1000000 nM T11615 D0D4CY 5336 IC50 > 1000000 nM T11615 D0L4VI 5862 Ki = 59000 nM T11615 D01IVR 11214940 IC50 = 200 nM T11615 C14GBL 76603 IC50 = 200000 nM T11615 C7BKY8 164701 IC50 = 26000 nM T11615 CUT07K 177491 IC50 = 35000 nM T11615 C2F6YX 299283 IC50 = 270000 nM T11615 CT5L2P 3086668 IC50 = 70000 nM T11615 C38RLF 4344716 IC50 = 150000 nM T11615 C8O9WI 6604711 IC50 > 1000000 nM T11615 CZLM83 19423375 IC50 > 1000000 nM T11615 CCF5P1 19423377 IC50 = 30000 nM T11615 CGXP45 19423407 IC50 = 900000 nM T11615 C7S6OA 19423412 IC50 = 700000 nM T11615 CBR97V 19423428 IC50 = 70000 nM T11615 C4F5IS 46200993 Ki = 117000 nM T11615 C14MZL 46229674 Ki = 52000 nM T11615 CO4PQ1 56662701 IC50 = 75000 nM T11615 CLSI08 56673081 IC50 = 920000 nM T11615 C2FQG0 56683051 IC50 > 1000000 nM T11615 CO1VE8 72710858 IC50 = 800 nM T11615 C4A2BO 72950385 IC50 = 60 nM T11615 CW7ZO4 91824786 IC50 = 30 nM T11615 CACN29 118247611 IC50 = 30 nM T11615 CT7H0F 118247614 IC50 = 100 nM T11615 CKXP79 118247618 IC50 = 300 nM T11615 CMDK86 118247619 IC50 = 10 nM T11615 C4LW6K 118247620 IC50 = 10 nM T11615 CEIN41 118247631 IC50 = 4 nM T11615 CU0Q1J 118247632 IC50 = 40 nM T11615 CQ2PV8 118247633 IC50 = 20 nM T11615 D06DUE 40539 IC50 = 5000 nM T11615 D0P3XO 5311459 IC50 = 5000 nM T46185 D01AZG 5073 Ki > 1000 nM T46185 D04JEE 4946 EC50 > 5011.87 nM T46185 D05SJW 6172 Ki = 467.74 nM T46185 D06HLY 5910 Ki = 12022.64 nM T46185 D08CTT 21855 Ki = 44.67 nM T46185 D09VBC 2562 Ki = 167 nM T46185 D09ZOQ 11519069 Ki = 0.15 nM T46185 D0B4TN 2381 Ki = 13.7 nM T46185 D0BZ7W 443879 Ki = 2.7 nM T46185 D0E6YQ 1935 Ki = 5800 nM T46185 D0G8NN 119570 Ki > 10000 nM T46185 D0H3HM 60795 Ki > 1000 nM T46185 D0H7KF 5002 Ki > 1000 nM T46185 D0L4YD 154059 Ki = 120.23 nM T46185 D0M0AM 11693 IC50 = 0.5012 nM T46185 D0M6VK 71183 Ki = 0.0631 nM T46185 D0Q9HF 187 EC50 = 7 nM T46185 D0RD5W 154417 Ki = 2.818 nM T46185 D0RG3O 174174 Ki = 0.344 nM T46185 D0T0LM 4848 Ki = 173.78 nM T46185 D0U7BW 5831 IC50 = 3.8 nM T46185 D0V4QS 135398745 Ki = 100 nM T46185 D0VP1V 11434515 IC50 < 0.03981 nM T46185 D0Y5AM 444031 Ki = 47 nM T46185 D0Z1RV 135398737 Ki = 100 nM T46185 D04YEW 25147683 IC50 = 97.3 nM T46185 D07EFM 2230 EC50 = 25 nM T46185 D09JLI 3009355 Ki > 10000 nM T46185 D0EY0A 42636350 IC50 = 80500 nM T46185 D0I5XU 16065403 Ki = 0.137 nM T46185 D0K4HW 135409468 Ki = 250 nM T46185 D0LI1C 44469321 IC50 > 10000 nM T46185 D0N1HW 5311200 Ki > 10000 nM T46185 D0R2OU 25070031 Ki = 3700 nM T46185 D0Z7AB 5487426 Ki = 0.49 nM T46185 D02JNY 10030021 Ki = 7.943 nM T46185 D05HKB 87934 EC50 = 400 nM T46185 D06ACX 6436265 Ki = 4.5 nM T46185 D06DZI 107780 Ki < 1000 nM T46185 D07IZF 9867750 Ki = 8 nM T46185 D08YVT 9894173 Ki = 0.89 nM T46185 D09FYQ 9577995 EC50 = 62.1 nM T46185 D0A2OW 107867 Ki = 52 nM T46185 D0J8UV 9928284 IC50 > 10000 nM T46185 D0PZ9R 45260374 Ki = 3.4 nM T46185 D0R1VL 132712 Ki = 30.2 nM T46185 D0UX0T 9571002 Ki = 1000 nM T46185 D0VZ3D 129989 Ki = 4.266 nM T46185 D0X8MZ 178030 EC50 = 296 nM T46185 C01PRU 1993 Ki = 59 nM T46185 C4AWJ9 2684 Ki = 851.14 nM T46185 C0H8GR 3191 IC50 > 1000 nM T46185 CKD46H 4022 Ki = 3235.94 nM T46185 C7VMZ3 4108 Ki = 2.399 nM T46185 CL53OW 6461 Ki = 0.68 nM T46185 C5H9CN 9287 Ki > 10000 nM T46185 C89UZB 18493 Ki = 1.54 nM T46185 CNZD18 36381 Ki = 835 nM T46185 CRCD50 60809 Ki = 8.128 nM T46185 C8E9XD 66007 IC50 = 18.6 nM T46185 C3WKC6 68835 IC50 > 100000 nM T46185 C3S8RF 71792 EC50 = 849 nM T46185 C6ZQ4D 72064 Ki = 1020 nM T46185 CA3W0P 100826 IC50 > 100000 nM T46185 CQA93V 118500 Ki = 1000 nM T46185 CN9W1S 129456 EC50 = 0.039 nM T46185 C27RUO 129486 Ki = 0.472 nM T46185 CG56JL 129993 Ki > 21000 nM T46185 C2WO0V 163938 IC50 = 20 nM T46185 CZ0UI5 208598 Ki = 20000 nM T46185 CHLK79 214124 Ki = 23.4 nM T46185 C71KVJ 275176 Ki = 281.5 nM T46185 CD65GI 315401 Ki = 5.38 nM T46185 C6OQ8S 410345 Ki = 15.1 nM T46185 CJ1QN5 425249 Ki = 5.85 nM T46185 C9R3VC 444015 Ki = 1.82 nM T46185 CW39FG 455656 Ki = 100 nM T46185 C91RPQ 455657 Ki = 100 nM T46185 CLU42H 456292 Ki = 760 nM T46185 CJKB92 456293 Ki = 485 nM T46185 CG48QX 456319 Ki = 35 nM T46185 C4AW8L 456611 Ki > 40 nM T46185 C2VJ3Z 456615 Ki = 0.8 nM T46185 CTU5D6 457875 Ki = 1323 nM T46185 CUWT43 461838 Ki = 352 nM T46185 C38ERL 461871 Ki > 1400 nM T46185 CHG02J 462395 Ki = 348 nM T46185 CU43EI 462571 Ki = 985 nM T46185 C47MIH 462573 Ki = 1678 nM T46185 CKI1S3 462772 Ki = 270 nM T46185 C9YW6M 462902 Ki = 164 nM T46185 CCHZ81 462989 Ki = 255 nM T46185 CF8X4A 463209 Ki = 68 nM T46185 CNVX67 463210 Ki = 169 nM T46185 C2HB4T 463319 Ki = 1225 nM T46185 CC85IE 463493 Ki = 31 nM T46185 C2T0PC 463502 Ki > 40 nM T46185 CH61SC 463517 Ki = 1 nM T46185 C8UQ6H 463616 Ki = 2031 nM T46185 CVQ5L9 463892 Ki = 202 nM T46185 CAP7I1 464036 Ki = 2500 nM T46185 CTB56C 474188 Ki = 1100 nM T46185 CZ49VF 474465 Ki = 497 nM T46185 C4J8NF 483747 Ki = 456 nM T46185 C7JQ2Z 502259 Ki = 613 nM T46185 CFJ63U 511332 Ki = 250 nM T46185 CX75UZ 598754 Ki > 19952.62 nM T46185 CC56KR 639794 Ki = 10471.29 nM T46185 C91GCI 657308 Ki = 0.413 nM T46185 CEGR96 657346 Ki = 1202.26 nM T46185 C04XRI 657347 Ki = 1202.26 nM T46185 CYO7F3 688566 IC50 = 0.4 nM T46185 CZN6S9 743974 EC50 > 15848.93 nM T46185 C08WCU 851833 Ki > 19952.62 nM T46185 CAX1I6 909982 Ki = 616.6 nM T46185 CO59NV 939077 IC50 = 2.83 nM T46185 CUD48J 952858 IC50 > 10000 nM T46185 CD97MX 1273944 Ki = 2238.72 nM T46185 CH5WR4 1421986 IC50 = 6900 nM T46185 CPL49A 2157678 EC50 > 30000 nM T46185 CTRP25 2396803 Ki = 794.33 nM T46185 CS8N5X 2736067 Ki = 7943.28 nM T46185 CUF0Z9 3009352 Ki = 4750 nM T46185 CMK58I 3009353 Ki = 4760 nM T46185 CPN54Q 3009354 Ki > 5700 nM T46185 C6ZYX5 3009356 Ki = 3512 nM T46185 C5X0LK 3009357 Ki > 6700 nM T46185 C91XVY 3233138 IC50 = 79.43 nM T46185 CJ6D8N 3342390 Ki < 1000 nM T46185 CI7DF6 3675988 Ki = 29512.09 nM T46185 CX3S8T 4715419 Ki = 4265.8 nM T46185 C12BJA 4995951 Ki = 537.03 nM T46185 CS71UA 5189681 IC50 > 30000 nM T46185 CR5LG3 5310989 IC50 = 4563.5 nM T46185 C1P3QG 5487543 EC50 = 26700 nM T46185 C07PJQ 6603753 Ki = 2089.3 nM T46185 C3A1FO 6604789 Ki = 50118.72 nM T46185 CFN7L4 6604866 Ki = 30.2 nM T46185 C2IP0Y 7022778 Ki = 107151.93 nM T46185 CVSC58 7047822 Ki = 77624.71 nM T46185 C32TSZ 7141654 Ki = 28840.32 nM T46185 C7NJZ2 7141656 Ki = 3235.94 nM T46185 CYH05F 9794266 Ki = 1200 nM T46185 CEDB68 9798900 IC50 = 14.5 nM T46185 CL94XF 9799291 Ki = 630 nM T46185 C8XGV3 9804849 IC50 = 480 nM T46185 C1P2KQ 9807612 Ki = 1.6 nM T46185 C7MBO3 9809330 Ki = 0.1259 nM T46185 CKR78B 9820835 EC50 = 1900 nM T46185 CMC3O6 9821459 Ki = 490 nM T46185 C6NJO3 9827782 Ki = 0.07 nM T46185 C80IET 9843967 Ki = 320 nM T46185 CH74OS 9846311 Ki = 530 nM T46185 C90VIH 9851621 Ki = 0.5 nM T46185 C3YI2L 9857572 IC50 = 22.9 nM T46185 CGO07X 9859365 Ki = 31 nM T46185 C1N0KW 9867847 Ki = 0.17 nM T46185 CU9Q4Y 9871136 Ki = 2.91 nM T46185 C14GTE 9871871 Ki = 2 nM T46185 C6EU0V 9872651 Ki = 1.1 nM T46185 CZHS28 9880462 Ki = 25 nM T46185 CJ5K1D 9889312 Ki = 2.7 nM T46185 CHK4U7 9894136 Ki = 6.9 nM T46185 CX4NP5 9894236 Ki = 0.2 nM T46185 CO4YW6 9894922 Ki = 15 nM T46185 CR5PO3 9903030 IC50 = 195.6 nM T46185 CUN81Q 9905249 Ki > 10000 nM T46185 C2U5LK 9905467 IC50 = 564.9 nM T46185 CF49JB 9905609 Ki > 1400 nM T46185 CCT20X 9905731 Ki = 6 nM T46185 CYWQ50 9906447 Ki = 462 nM T46185 CDB9E1 9909907 Ki = 15.85 nM T46185 CL5HA4 9910802 Ki = 460 nM T46185 CXAV92 9911615 Ki = 3801.89 nM T46185 CXAY37 9913341 IC50 = 0.5012 nM T46185 C24PKZ 9913892 Ki = 316.23 nM T46185 CB3LH7 9916852 Ki = 0.01 nM T46185 CG4PD5 9927975 EC50 = 2 nM T46185 C3L5GV 9928017 IC50 = 1.8 nM T46185 CRV17M 9931930 Ki = 1071.52 nM T46185 C50NSR 9936450 Ki = 3.162 nM T46185 CCUW90 9937474 Ki = 0.1995 nM T46185 C0HR4G 9938599 Ki = 1 nM T46185 C65PMK 9944783 IC50 = 13.6 nM T46185 C36NIB 9946010 IC50 = 4.7 nM T46185 CKQM18 9946298 Ki = 0.79 nM T46185 CY4L1D 9946632 IC50 = 115.7 nM T46185 CUCT38 9948957 Ki = 844 nM T46185 C7TD1E 9953227 Ki = 0.37 nM T46185 CFG21X 9966959 IC50 = 76.2 nM T46185 CH23EP 9967590 IC50 = 3.7 nM T46185 CYNT43 9968046 Ki = 169.82 nM T46185 CQF52V 9969695 Ki = 158.49 nM T46185 CCM72P 9974222 IC50 = 243.6 nM T46185 CT26UJ 9974229 Ki = 51 nM T46185 C6QZ8W 9984928 Ki = 0.16 nM T46185 C3G0VC 9985181 Ki = 32 nM T46185 C9XS0E 9990434 IC50 = 2840 nM T46185 CD9A5M 9991939 Ki = 270 nM T46185 C8F4XT 9991979 Ki = 600 nM T46185 CYK1U4 9996901 IC50 = 229.6 nM T46185 C9FR0C 9998508 Ki = 416.87 nM T46185 CQL12P 10004545 Ki > 2000 nM T46185 CK19GL 10007637 IC50 = 0.6 nM T46185 C7GSR4 10009225 EC50 = 46.77 nM T46185 CGY8P7 10009554 Ki = 0.51 nM T46185 CQP9F4 10012808 EC50 > 51000 nM T46185 CV0KA3 10019339 EC50 = 683 nM T46185 CV7R9F 10020040 Ki > 10000 nM T46185 C6V3NE 10020614 Ki = 145 nM T46185 CQZ0K4 10027177 EC50 > 50000 nM T46185 C7I6DA 10035281 Ki = 2700 nM T46185 CO69GW 10035533 IC50 = 519 nM T46185 CBJ63D 10043954 Ki = 323.59 nM T46185 CPCL60 10044685 Ki = 316.23 nM T46185 CQ8F9I 10049361 Ki = 5.012 nM T46185 C56FEU 10053613 IC50 = 4.8 nM T46185 C9Z3TI 10058347 IC50 = 519 nM T46185 C2WJS1 10058649 Ki = 330 nM T46185 CORA81 10058744 IC50 = 6010 nM T46185 CV6A5I 10061123 Ki = 2200 nM T46185 C9OQ2S 10066369 Ki = 25.12 nM T46185 CI6SD7 10066972 Ki = 331.13 nM T46185 C1GUM0 10080742 IC50 = 10800 nM T46185 C6Z5CY 10081053 IC50 = 4460 nM T46185 CCO72H 10082470 IC50 = 480 nM T46185 CQ3O0X 10085070 IC50 = 7930 nM T46185 C8NQ3I 10092649 Ki = 320 nM T46185 C2GZC9 10096939 Ki = 1.6 nM T46185 C4IZ5H 10101246 Ki = 0.2291 nM T46185 CT4XE6 10103909 Ki = 2800 nM T46185 CO0V4J 10104047 EC50 = 680 nM T46185 CHUE04 10104527 Ki > 18000 nM T46185 COR41M 10105880 Ki = 9200 nM T46185 CU25MW 10109130 Ki = 0.2 nM T46185 CIN03S 10109563 Ki = 2.512 nM T46185 CG0O9Z 10109893 IC50 = 7.943 nM T46185 CUT05R 10114698 Ki = 7244.36 nM T46185 CS10UG 10119364 Ki = 1.3 nM T46185 C9XDU8 10119938 IC50 = 3.2 nM T46185 C20GMN 10132599 IC50 = 42.1 nM T46185 CFH60N 10133281 IC50 = 22.7 nM T46185 C90FZG 10139614 Ki = 4570.88 nM T46185 C0PO3J 10142923 IC50 = 0.5012 nM T46185 CPF96U 10143717 IC50 = 1.1 nM T46185 CC8YJ1 10143857 IC50 = 8.4 nM T46185 C7LP4V 10143953 IC50 = 1.01 nM T46185 CYU79M 10143955 Ki = 0.06 nM T46185 C9DY4P 10155225 Ki = 6.31 nM T46185 CDOI12 10155850 Ki = 19.95 nM T46185 CG78WP 10160073 Ki = 338.84 nM T46185 CZ8E9X 10160219 Ki = 1445.44 nM T46185 C4G8OW 10163651 Ki = 0.89 nM T46185 CVI4O6 10164136 IC50 = 8.9 nM T46185 CR1DZ8 10164480 Ki = 32 nM T46185 CXCT70 10165876 IC50 = 1.6 nM T46185 C4TR5Q 10180872 Ki = 1 nM T46185 C1B8RO 10187215 IC50 = 7.6 nM T46185 CO05SP 10199963 Ki = 5 nM T46185 COR14Y 10203251 Ki = 512.86 nM T46185 CB69ND 10204457 Ki = 7.3 nM T46185 CUW93D 10208896 IC50 = 4 nM T46185 C57WMS 10208971 IC50 = 3.9 nM T46185 C2H1WR 10220392 IC50 = 25800 nM T46185 CJ5V2S 10225340 Ki = 3.07 nM T46185 C04QCB 10225881 Ki = 2187.76 nM T46185 C6A5KD 10226456 Ki = 15.85 nM T46185 C8XY5N 10229166 IC50 = 10.9 nM T46185 CHX43K 10230930 Ki = 0.17 nM T46185 CO64WJ 10236758 Ki = 204.17 nM T46185 CRQ8D4 10240891 IC50 = 7890 nM T46185 CE69PK 10242813 Ki = 400 nM T46185 CQB1O6 10243426 Ki = 96 nM T46185 CEYJ57 10244370 Ki = 3000 nM T46185 C49MUR 10246307 IC50 = 4.2 nM T46185 C3W2YB 10248541 IC50 = 960 nM T46185 C3QGA5 10251795 EC50 > 50000 nM T46185 CW90FO 10261985 EC50 = 6.7 nM T46185 CLS61Z 10262405 IC50 = 20600 nM T46185 C1FCP7 10262466 Ki = 70 nM T46185 CH31DX 10267394 Ki > 10000 nM T46185 CC6RP7 10267601 IC50 = 255.2 nM T46185 CT07QH 10269503 Ki = 1.585 nM T46185 CFN5O4 10269504 Ki = 20 nM T46185 CCN9B4 10269809 Ki = 39.81 nM T46185 CY3E5J 10274019 Ki = 0.14 nM T46185 C7CYM8 10275847 Ki = 1.3 nM T46185 C8HD7O 10291366 Ki = 0.79 nM T46185 C6N9XM 10291977 Ki = 0.4 nM T46185 CG6I4F 10299489 Ki = 5 nM T46185 C7WMZ6 10300660 IC50 = 17.7 nM T46185 CCD1L2 10302719 Ki = 9.6 nM T46185 CU89JD 10314060 Ki > 10000 nM T46185 CD1C0H 10315426 Ki = 309.03 nM T46185 CF05IP 10324012 Ki = 0.26 nM T46185 CWP67J 10330721 Ki > 18000 nM T46185 CLW9R8 10330893 Ki = 410 nM T46185 CYIS62 10333583 IC50 = 4010 nM T46185 C3E5CB 10337773 Ki = 50118.72 nM T46185 C9YR5B 10339062 Ki = 1100 nM T46185 CV0BU1 10348407 EC50 = 54.95 nM T46185 C6S7GK 10354348 IC50 = 100000 nM T46185 C5M9WO 10354430 Ki = 2700 nM T46185 C5UTA9 10356006 IC50 = 20600 nM T46185 CP0LR5 10357756 Ki > 10000 nM T46185 C7BZ1R 10358345 IC50 = 227 nM T46185 CBSA40 10360219 Ki = 95.5 nM T46185 CLM8P2 10365639 Ki = 4.49 nM T46185 C9LWG3 10369004 IC50 > 1000 nM T46185 CLHJ56 10375002 EC50 = 270 nM T46185 CY9G0R 10375322 IC50 = 8600 nM T46185 CUD07Z 10376012 IC50 = 5080 nM T46185 CXN2K4 10376182 IC50 = 9650 nM T46185 C72EML 10392704 IC50 = 91.5 nM T46185 CR1EA3 10393100 Ki = 0.7 nM T46185 C85QEA 10397133 IC50 = 1040 nM T46185 C5TX2E 10397356 IC50 = 1700 nM T46185 CUBA69 10398843 Ki = 200 nM T46185 CQW10P 10399393 IC50 = 2180 nM T46185 C30DKF 10405613 Ki = 71.2 nM T46185 CPMI73 10417432 Ki = 0.51 nM T46185 CALE73 10419574 IC50 = 3980 nM T46185 CID42C 10420458 IC50 = 1900 nM T46185 C0IPX1 10421689 Ki = 990 nM T46185 CL7D2U 10421982 Ki = 260 nM T46185 C07QHE 10429011 Ki = 460 nM T46185 CE3MX5 10437400 Ki = 1.1 nM T46185 C5BEJ0 10442081 EC50 = 43 nM T46185 CIRS06 10442337 EC50 = 41 nM T46185 CS63AC 10447114 Ki > 10000 nM T46185 CAW4U0 10451242 EC50 = 1655 nM T46185 CA3CY4 10451634 Ki = 97 nM T46185 C4C7UG 10457079 Ki = 0.07586 nM T46185 C4GBW9 10461523 Ki = 0.1 nM T46185 CI8R9A 10465050 Ki = 1900 nM T46185 C6B5DJ 10465524 IC50 = 15900 nM T46185 CK9ZH7 10466231 Ki = 99 nM T46185 CVK48E 10467755 Ki = 4200 nM T46185 C53SCK 10468535 Ki = 98 nM T46185 CE6JH3 10473919 Ki = 692 nM T46185 C26BIM 10475156 Ki = 5500 nM T46185 CEF2O6 10478367 Ki > 10000 nM T46185 C1GT3O 10487582 IC50 = 610 nM T46185 C8COH6 10499832 IC50 = 661.1 nM T46185 C18ZYN 10500741 Ki = 30 nM T46185 CU0B8N 10501523 Ki = 37000 nM T46185 CO62HL 10503358 Ki = 310 nM T46185 CS1P4M 10511551 IC50 = 700 nM T46185 CKP8N1 10515352 IC50 = 20800 nM T46185 CP9M5J 10516408 IC50 = 1668.5 nM T46185 C37PDA 10518821 IC50 = 14598.2 nM T46185 C6T1JW 10521205 IC50 = 1944.1 nM T46185 C4WZ3R 10522202 IC50 = 468 nM T46185 C5MB2F 10522336 IC50 = 486.1 nM T46185 C3EZ5Y 10525412 Ki = 22 nM T46185 C0K9HN 10538337 IC50 = 28264.5 nM T46185 CD9RI5 10539130 IC50 = 27200 nM T46185 C3Y6JB 10546275 IC50 = 22.2 nM T46185 CI3GQ6 10547222 IC50 = 1174.8 nM T46185 C6XKZ9 10549581 IC50 = 475 nM T46185 CSC81Z 10551354 Ki = 480 nM T46185 CUJ3W9 10563152 IC50 = 47900 nM T46185 CFD40Z 10567192 IC50 = 273.5 nM T46185 C4AL8Q 10569816 IC50 = 956.4 nM T46185 CHI03M 10572657 Ki = 4600 nM T46185 C0Z5PY 10572658 Ki = 6400 nM T46185 CV62YH 10573458 Ki = 2400 nM T46185 CB37SH 10573693 IC50 = 2573.4 nM T46185 CR2GX4 10574041 Ki = 8600 nM T46185 C71VMD 10591874 IC50 = 450.6 nM T46185 C94VUE 10592484 IC50 = 748.5 nM T46185 C51LBK 10593954 IC50 = 2213.8 nM T46185 CH2QU8 10594386 IC50 = 10943.7 nM T46185 CY54RA 10595006 Ki = 1100 nM T46185 C6VGM0 10597259 Ki = 1300 nM T46185 CVY63G 10598540 Ki = 9400 nM T46185 CZRJ60 10610375 IC50 = 1727.9 nM T46185 C5HKT1 10610448 IC50 = 8900 nM T46185 CX01SE 10611310 IC50 = 394.8 nM T46185 CO3H7D 10614695 IC50 = 954.3 nM T46185 C3BK2J 10619926 Ki = 1800 nM T46185 C34LMA 10621363 Ki = 70 nM T46185 CSGO98 10622033 Ki = 2000 nM T46185 C92HRJ 10622718 Ki = 21000 nM T46185 CLJ29W 10623721 Ki = 3400 nM T46185 CJL4R1 10636001 IC50 = 542.3 nM T46185 C09XHV 10638050 IC50 = 1500.6 nM T46185 C5VWL8 10641009 IC50 = 238.2 nM T46185 C2ZTE6 10646906 Ki = 220 nM T46185 CDAG26 10646948 Ki = 37 nM T46185 CZ7M1D 10647553 Ki = 6900 nM T46185 CX49UY 10647703 Ki = 310 nM T46185 CONH15 10663572 IC50 = 241.3 nM T46185 C6WQ2Z 10664532 IC50 = 1480.7 nM T46185 C8CF4H 10666533 IC50 = 734.6 nM T46185 C56EGM 10670917 Ki = 330 nM T46185 C1DSK6 10670961 Ki = 930 nM T46185 CUYW18 10671167 Ki = 17000 nM T46185 C0AV8X 10678449 IC50 = 220 nM T46185 C32KQX 10684720 IC50 = 1865.1 nM T46185 CZQY38 10686494 EC50 = 240 nM T46185 C32EGP 10686988 IC50 = 405 nM T46185 C9O6LN 10688349 IC50 = 4496.8 nM T46185 C6PDH5 10693031 Ki = 24 nM T46185 CW91HU 10707175 IC50 = 69300 nM T46185 C62MCG 10716120 Ki = 2300 nM T46185 CS3W1G 10718110 Ki = 17000 nM T46185 CEB3A5 10726038 IC50 = 240 nM T46185 C5OF4K 10739662 Ki = 3300 nM T46185 CC21XD 10755732 IC50 = 470.7 nM T46185 CHL29Z 10755733 IC50 = 427.5 nM T46185 C4JXA3 10757736 IC50 = 1611.2 nM T46185 C15WSV 10759971 Ki = 13.3 nM T46185 CPQ7Z3 10760249 IC50 = 136 nM T46185 C5P3DQ 10761219 IC50 = 3323.1 nM T46185 CTNG89 10777343 IC50 = 38600 nM T46185 CX4LT3 10777692 IC50 = 2763.7 nM T46185 CC7TL1 10778462 IC50 = 84400 nM T46185 CU5SO1 10778750 IC50 = 24700 nM T46185 CA4QI2 10782321 IC50 = 10788.8 nM T46185 C4N9IT 10782462 IC50 = 666.3 nM T46185 C6FC0M 10784004 IC50 = 1035.2 nM T46185 CV8TE0 10785471 IC50 = 20.5 nM T46185 CLI6Z3 10789183 Ki = 19.95 nM T46185 CW5TJ6 10797864 IC50 = 31 nM T46185 C9SEA6 10806268 IC50 = 73.3 nM T46185 CGR64V 10808719 IC50 = 2162.1 nM T46185 C3QK4R 10810094 Ki = 14000 nM T46185 CR4XK8 10812455 Ki = 260 nM T46185 CX9B7I 10826990 IC50 = 46600 nM T46185 CK1D3J 10827157 IC50 = 1248.2 nM T46185 CR1X5L 10829928 IC50 = 1222.1 nM T46185 C0GS8Z 10830843 Ki = 15000 nM T46185 C2M0QO 10834711 Ki = 79 nM T46185 C27NPT 10835518 Ki = 3100 nM T46185 C2S6DG 10836338 Ki = 2400 nM T46185 CB7E2O 10846833 IC50 = 2200 nM T46185 CFQ74S 10848032 IC50 = 15200 nM T46185 CH9WK6 10851853 IC50 = 600.7 nM T46185 CX6AP3 10852843 IC50 = 4100.3 nM T46185 C5PRT6 10854879 IC50 = 773.5 nM T46185 C8HI5L 10854880 IC50 = 52.5 nM T46185 CZ85AJ 10862395 Ki = 1348.96 nM T46185 CHE9P4 10865439 Ki = 9.2 nM T46185 CMS71D 10865495 EC50 = 134.9 nM T46185 CCM3L9 10870954 Ki = 14791.08 nM T46185 C2YNC5 10871551 Ki = 107.15 nM T46185 CFAD04 10874119 Ki = 1348.96 nM T46185 CTV95B 10880435 Ki = 234.42 nM T46185 C4A8QE 10916286 Ki = 2454.71 nM T46185 CQLR32 10919522 Ki = 0.82 nM T46185 CC12TE 10925451 Ki = 363.08 nM T46185 CU09AV 10937901 IC50 = 518 nM T46185 C5LVY0 10949838 Ki = 707.95 nM T46185 CE05FM 10951142 Ki = 371.54 nM T46185 C3K6JV 10957754 Ki = 263.03 nM T46185 CN4QT5 10963509 Ki = 8.6 nM T46185 C4WV8L 10969390 Ki = 32.36 nM T46185 CTYZ13 10969696 Ki = 1445.44 nM T46185 C8LWG4 10974720 EC50 = 177.83 nM T46185 C41PXY 10982070 Ki = 416.87 nM T46185 C9E2MP 10984804 Ki = 3100 nM T46185 CW0HB1 10985526 EC50 = 70.79 nM T46185 C2W3GM 11000399 Ki = 6760.83 nM T46185 C6NH9T 11001809 Ki = 6025.6 nM T46185 CQ8D4K 11004046 Ki = 512.86 nM T46185 C6BG1N 11006792 Ki = 13 nM T46185 CU4Z0J 11011332 Ki = 5370.32 nM T46185 CZK86F 11011757 Ki = 257.04 nM T46185 CVA6U9 11012653 Ki = 144.54 nM T46185 CPM1Z7 11012712 Ki = 1071.52 nM T46185 CW23BJ 11013666 Ki = 229.09 nM T46185 C6TF5I 11015312 Ki = 2344.23 nM T46185 C7Y1DO 11024241 Ki = 912.01 nM T46185 C3L9ON 11034265 Ki = 112.2 nM T46185 CHDT49 11039424 Ki = 30 nM T46185 CP9OJ6 11045444 Ki = 676.08 nM T46185 C4ZUH9 11048067 Ki = 218.78 nM T46185 CQ8O3Y 11057942 Ki > 26915.35 nM T46185 CIG31V 11061341 Ki = 12 nM T46185 CT3XN5 11071537 Ki = 15.85 nM T46185 C5VQ6H 11079969 Ki = 1071.52 nM T46185 CWS56C 11092603 Ki = 239.88 nM T46185 C02MPO 11099206 Ki = 398.11 nM T46185 CSNA03 11101362 Ki = 3235.94 nM T46185 CF81CB 11110049 Ki = 93325.43 nM T46185 C7ROJ1 11112362 Ki = 5370.32 nM T46185 C9CY0M 11120347 Ki = 588.84 nM T46185 CD20CQ 11120503 EC50 = 1096 nM T46185 C2C4AN 11131099 Ki = 1023.29 nM T46185 C1T9WI 11143997 Ki = 2187.76 nM T46185 C34JRO 11169365 Ki = 630.96 nM T46185 CX69QO 11223597 Ki = 0.73 nM T46185 CI1EN4 11306851 IC50 = 4.5 nM T46185 CBR60Z 11318734 IC50 > 3162.28 nM T46185 C85LYP 11430418 IC50 > 1000 nM T46185 C9FNM4 11431811 Ki = 0.01995 nM T46185 CGD57K 11431873 Ki = 0.1 nM T46185 C9NUV4 11442477 IC50 = 7.2 nM T46185 CIN42A 11489418 IC50 = 0.36 nM T46185 CTVZ02 11503335 IC50 = 13.8 nM T46185 CBZ5E8 11508710 IC50 = 26.5 nM T46185 CSP02B 11510357 IC50 = 53.7 nM T46185 CGCF61 11515738 Ki = 51286.14 nM T46185 C7OKD1 11518067 IC50 = 12.5 nM T46185 CY63VP 11523050 Ki = 15488.17 nM T46185 C07AJD 11530306 Ki = 28840.32 nM T46185 C8UB7G 11531643 Ki = 6.166 nM T46185 CQ08DH 11539632 IC50 = 4.5 nM T46185 CWUP85 11542982 Ki < 100000 nM T46185 C6B2XK 11547052 IC50 = 55.9 nM T46185 CNZJ38 11552174 IC50 = 39.1 nM T46185 CP9UJ1 11569907 IC50 = 1.82 nM T46185 CP04FM 11569925 IC50 = 50.9 nM T46185 CYW90N 11583261 IC50 = 30.2 nM T46185 C6D1MA 11584660 IC50 = 316.23 nM T46185 CEHP14 11586481 Ki < 100000 nM T46185 CP3Y7J 11588240 Ki = 77624.71 nM T46185 CP3G5L 11602980 IC50 = 19.6 nM T46185 C15DMA 11617374 IC50 = 90.7 nM T46185 CE07UT 11619197 IC50 = 48 nM T46185 CQ5PI4 11622544 Ki < 100000 nM T46185 CK4GS9 11626846 IC50 = 34.7 nM T46185 CF2ZC0 11651360 Ki < 100000 nM T46185 CHKN81 11653111 Ki = 9332.54 nM T46185 C27XOS 11660220 Ki < 100000 nM T46185 C0N4BQ 11672895 Ki = 87096.36 nM T46185 C0ZK8U 11678377 IC50 = 29.8 nM T46185 CN4Z5C 11679149 IC50 > 10000 nM T46185 CI5B1R 11690967 IC50 = 10.9 nM T46185 CQD96L 11691949 Ki = 0.94 nM T46185 CW8CE2 11694118 Ki < 100000 nM T46185 CF8MO2 11694119 Ki = 89125.09 nM T46185 CMT6F0 11695697 IC50 = 347.6 nM T46185 CY31MF 11712407 IC50 = 60.8 nM T46185 C9BF1S 11715398 Ki < 100000 nM T46185 CWE71N 11718536 Ki = 80.1 nM T46185 C0E9SG 11725107 EC50 = 2690 nM T46185 C0O2QC 11725334 IC50 = 1.7 nM T46185 CEY7J3 11729182 Ki = 4073.8 nM T46185 CPG15O 11743399 IC50 > 1000 nM T46185 C4QVR6 11748799 Ki = 15.49 nM T46185 CQLP36 11759058 Ki = 39810.72 nM T46185 CW3GA7 11759212 Ki = 33.11 nM T46185 CBM05D 11759379 Ki = 851.14 nM T46185 CFZ4L5 11767229 Ki = 72 nM T46185 C39HRB 11793999 IC50 = 120.7 nM T46185 CM16WE 11794901 Ki = 320 nM T46185 CT8P7Q 11796409 Ki = 1400 nM T46185 C91DQM 11796509 Ki = 270 nM T46185 CHEA80 11798126 Ki = 1000 nM T46185 CT4F2C 11808040 Ki = 12.3 nM T46185 CXQ10I 11808946 Ki = 97.72 nM T46185 C6EXD3 11808947 Ki = 51.29 nM T46185 C30WRH 11809446 Ki = 4897.79 nM T46185 CN9M8E 11811722 IC50 = 4540 nM T46185 CF1S7Q 11819427 IC50 = 3150 nM T46185 C3MQW7 11819545 Ki = 1700 nM T46185 CQW16Z 11819782 Ki = 5011.87 nM T46185 C0BPK3 11819882 Ki = 620 nM T46185 C2KW3U 11819883 Ki = 1700 nM T46185 CJIA51 11828362 Ki = 44 nM T46185 C0QKL8 11828771 EC50 = 36.31 nM T46185 CR9FJ2 11833737 Ki = 1949.84 nM T46185 CZ3AX9 11834199 Ki = 44.67 nM T46185 C8JQL7 11957735 IC50 > 10000 nM T46185 CL91TM 11968014 Ki = 3.02 nM T46185 C5P3XD 12586122 EC50 = 18000 nM T46185 CYU4P5 12739458 Ki = 4304 nM T46185 CR10FQ 13567080 Ki = 7.586 nM T46185 COT9Z6 13981863 Ki = 0.45 nM T46185 C1IDP8 13981864 Ki = 2.52 nM T46185 CPX7C8 14210083 Ki = 1.738 nM T46185 C19BYU 14479864 IC50 < 1 nM T46185 CS54WY 14537188 Ki = 0.165 nM T46185 CA87RQ 14660293 IC50 = 6700 nM T46185 CU36CN 14685523 Ki = 1500 nM T46185 CMO81H 14925759 Ki = 16595.87 nM T46185 CVNK57 15065550 Ki = 102.33 nM T46185 CZS96E 15105207 Ki = 4900 nM T46185 C38UHI 15105209 Ki = 2271 nM T46185 C49DYR 15105211 Ki = 1569 nM T46185 CZ16XJ 15157137 Ki = 26.9 nM T46185 C5VC9Z 15157138 Ki = 19.7 nM T46185 C7VT5X 15157139 Ki = 258 nM T46185 CD3MI7 15157140 Ki = 248 nM T46185 CY80DC 15157141 Ki = 246 nM T46185 CAF40B 15181802 IC50 = 7300 nM T46185 CSA5Y2 15196231 Ki > 53000 nM T46185 CO4EB0 15196232 Ki = 27000 nM T46185 COIG73 15196233 Ki = 15900 nM T46185 C80ICP 15196234 Ki = 390 nM T46185 CIV27H 15196235 Ki = 5000 nM T46185 CXZB18 15196236 Ki = 160 nM T46185 CEH60Q 15196354 Ki = 1300 nM T46185 CN1RW5 15392110 Ki = 0.2 nM T46185 CD9BL8 15407072 Ki = 9 nM T46185 CP7JQ0 15407073 Ki = 0.6 nM T46185 C36USC 15407074 Ki = 0.2 nM T46185 CW2VN5 15407088 Ki = 0.13 nM T46185 CMK9G7 15407089 Ki = 0.073 nM T46185 CEOD62 15453419 Ki = 0.11 nM T46185 C4B1VS 15463387 Ki = 0.3 nM T46185 CC2DK3 15463388 Ki = 0.15 nM T46185 C9C6WP 15629515 Ki > 50000 nM T46185 C4PYE0 15681299 IC50 = 1630 nM T46185 C48IJQ 15681300 IC50 = 5280 nM T46185 C0T6NK 15681301 IC50 = 15590 nM T46185 CG0RN6 15681303 IC50 = 59300 nM T46185 CEW1M8 15749863 Ki = 30000 nM T46185 CJ5Z9T 15749864 Ki = 50000 nM T46185 C9Y8AF 15870384 Ki = 0.4 nM T46185 CH85WD 15870389 Ki = 12 nM T46185 CIW40C 15888010 Ki = 240 nM T46185 CJKM40 15888011 Ki = 11 nM T46185 CT64BE 15945874 IC50 = 158.49 nM T46185 CG8KR9 16005860 IC50 = 8000 nM T46185 CUB5X2 16038385 EC50 = 630.96 nM T46185 CL1CM4 16065135 Ki = 1.6 nM T46185 CI1QH2 16065136 Ki = 12 nM T46185 CCS3K1 16065268 Ki = 2.6 nM T46185 CVZ68N 16065402 Ki = 0.056 nM T46185 CZ47FJ 16071018 EC50 = 630.96 nM T46185 C3T0UX 16085999 Ki = 220 nM T46185 CWI32N 16086000 Ki = 730 nM T46185 C71HBL 16086001 Ki = 73 nM T46185 C7EM1G 16086003 Ki = 3000 nM T46185 CFU72Z 16086004 Ki = 3700 nM T46185 CTOM27 16086005 Ki = 94 nM T46185 C7WF9Y 16086059 Ki = 490 nM T46185 C05YVJ 16086060 Ki = 450 nM T46185 CMQ8U3 16086061 Ki = 1300 nM T46185 CEI8G1 16086062 Ki = 68 nM T46185 CGB89M 16086063 Ki = 19 nM T46185 CUS73E 16086064 Ki = 110 nM T46185 CHJ07L 16086065 Ki = 1200 nM T46185 CEV68D 16086066 Ki = 310 nM T46185 CIX9M7 16086067 Ki = 100 nM T46185 C1XZ7V 16094783 Ki = 39.81 nM T46185 CO16DS 16094788 Ki = 2.512 nM T46185 CYN71L 16094791 Ki = 39.81 nM T46185 C2HK7W 16094793 Ki = 63.1 nM T46185 C9R0JN 16094810 Ki = 158.49 nM T46185 CTYI57 16115796 Ki = 2.754 nM T46185 C5HSD9 16115797 Ki = 1.072 nM T46185 CQ85FK 16115798 Ki = 4.266 nM T46185 CR1Z4N 16115799 Ki = 4.467 nM T46185 CLA6E0 16115800 Ki = 3.388 nM T46185 CTE0R7 16115942 Ki = 1.479 nM T46185 C7IC9E 16115944 Ki = 0.7762 nM T46185 CQ3C9X 16115946 Ki = 0.8318 nM T46185 C0JGY1 16115950 Ki = 4.898 nM T46185 CZ67DO 16115951 Ki = 2.754 nM T46185 CO3YU4 16116082 Ki = 0.4677 nM T46185 C3IKJ0 16116084 Ki = 0.955 nM T46185 CWU6P3 16123945 EC50 = 630.96 nM T46185 C6B4YR 16124705 Ki = 515 nM T46185 C42YXI 16124706 Ki = 107 nM T46185 CY0KP2 16124707 Ki = 187 nM T46185 C7RN3Z 16124708 Ki = 520 nM T46185 C8RVY4 16124710 Ki = 908 nM T46185 CZ7JF4 16124769 Ki = 629 nM T46185 CI1G8P 16125223 Ki = 82.2 nM T46185 CRW9N0 16125257 Ki = 1810 nM T46185 CK1OD5 16125325 Ki = 862 nM T46185 CXY50Q 16125331 Ki = 0.73 nM T46185 CA05KV 16125335 Ki = 27.4 nM T46185 C5G6IH 16125370 Ki = 2 nM T46185 CGUF57 16125371 Ki = 2272 nM T46185 C0J6CH 16125372 Ki = 207 nM T46185 C9YJT7 16125373 Ki = 73.3 nM T46185 C75NYZ 16125374 Ki = 96.8 nM T46185 CN5LU9 16125398 Ki = 157 nM T46185 CNHJ78 16125400 Ki = 108 nM T46185 CP31TE 16125437 Ki = 2952 nM T46185 CD9NV1 16125443 Ki = 2918 nM T46185 CE8G4T 16125505 Ki = 411 nM T46185 CVA18O 16125506 Ki = 1681 nM T46185 CQV41Z 16125507 Ki = 328 nM T46185 CR0K3N 16125508 Ki = 302 nM T46185 CS51VQ 16125509 Ki = 927 nM T46185 CKBU51 16125529 Ki = 2010 nM T46185 CA32GJ 16125531 Ki = 884 nM T46185 C1IC0F 16125541 Ki = 1.66 nM T46185 C29GWL 16125567 Ki = 328 nM T46185 CV03SP 16125568 Ki = 296 nM T46185 CXE2Y7 16125571 Ki = 695 nM T46185 C2AUB0 16125585 Ki = 47.8 nM T46185 C52IGT 16125587 Ki = 8.84 nM T46185 C8EH5G 16125589 Ki = 31.5 nM T46185 CFNB10 16125591 Ki = 9.92 nM T46185 CZ51NP 16125593 Ki = 1152 nM T46185 CW3U7K 16125618 Ki = 490 nM T46185 C3AI6K 16125619 Ki = 47.9 nM T46185 CG4AD1 16125620 Ki = 225 nM T46185 CR8BD3 16125621 Ki = 182 nM T46185 CIN56P 16125640 Ki = 552 nM T46185 CB5MC6 16125642 Ki = 2.39 nM T46185 CPM1Z9 16125646 Ki = 94.5 nM T46185 C81PZO 16125648 Ki = 1014 nM T46185 C91FGA 16125680 Ki = 302 nM T46185 CMN0P3 16125681 Ki = 955 nM T46185 C4BYI2 16125682 Ki = 1141 nM T46185 C1M2KX 16125683 Ki = 166 nM T46185 C91OQV 16125698 Ki = 268 nM T46185 CO02CS 16125704 Ki = 88.5 nM T46185 CZ2IS9 16660294 Ki > 10000 nM T46185 CEA26S 16664965 Ki = 21.9 nM T46185 CO1W8M 16721019 Ki = 1.8 nM T46185 CDB83R 17516658 EC50 > 30000 nM T46185 C45VOE 18342968 Ki = 40 nM T46185 C7T8JC 19958494 Ki > 10000 nM T46185 C6LI5E 19958507 Ki > 10000 nM T46185 C3T5HF 21509921 Ki > 10000 nM T46185 C4FNZ8 21862266 Ki = 9700 nM T46185 CBN84K 22065997 Ki > 10000 nM T46185 C5WCD3 22745278 EC50 = 11.9 nM T46185 C3IQT5 23352279 Ki = 1550 nM T46185 C5SUY3 23352285 Ki = 2600 nM T46185 C5Y1MK 23983764 Ki = 3.631 nM T46185 CL4WV2 24180125 IC50 = 6280 nM T46185 CXCO68 24192587 Ki = 348 nM T46185 C8KTP0 24739387 IC50 = 10000 nM T46185 C70CVK 24739554 IC50 > 10000 nM T46185 CSDA50 24739886 IC50 = 2000 nM T46185 C7I4LK 24750278 IC50 = 150 nM T46185 CY21RE 24841480 Ki = 100 nM T46185 C4SY8G 24846938 Ki = 7.93 nM T46185 CF26NI 24865894 Ki = 1258.93 nM T46185 CJ4FM6 24865895 Ki = 37153.52 nM T46185 C20VHK 24871823 IC50 = 7000 nM T46185 C43RTZ 24882193 IC50 = 3200 nM T46185 C9YN3A 24894514 Ki = 30902.95 nM T46185 C8ND1U 24894515 Ki = 47863.01 nM T46185 CX2HR8 24894516 Ki = 15848.93 nM T46185 CG4B9R 24894624 Ki = 7413.1 nM T46185 C7KF9R 24894626 Ki = 1659.59 nM T46185 CFA60S 24894627 Ki = 3715.35 nM T46185 CT8B3K 24894629 Ki = 1905.46 nM T46185 CMF04K 24894631 Ki = 41686.94 nM T46185 CP08SJ 24894632 Ki = 14454.4 nM T46185 CLJK58 24894633 Ki = 19498.45 nM T46185 CR86FA 24894634 Ki = 14125.38 nM T46185 C9J3NX 24894636 Ki = 2691.53 nM T46185 CUY89J 24936155 Ki = 280 nM T46185 CR7D1L 24967746 EC50 = 19.95 nM T46185 CFDQ56 24996645 IC50 = 340 nM T46185 CT93PZ 25010559 Ki = 3.162 nM T46185 C5MYC3 25010776 EC50 > 30000 nM T46185 C1VRJ3 25014630 IC50 = 3600 nM T46185 C18VYH 25015647 EC50 > 40000 nM T46185 CA20NZ 25025581 Ki = 199.53 nM T46185 C8JW9U 25034110 IC50 = 5011.87 nM T46185 C9OC1I 25034111 IC50 = 125.89 nM T46185 C3DB4P 25034112 IC50 = 19952.62 nM T46185 CH67WY 25034180 IC50 = 1584.89 nM T46185 CXBF68 25110764 EC50 > 50000 nM T46185 C50IKG 25110765 EC50 > 50000 nM T46185 CK0BT7 25147647 Ki = 1000 nM T46185 CE2OG1 25199525 EC50 > 15848.93 nM T46185 CRFJ43 25207745 EC50 = 2511.89 nM T46185 CP2T6G 25230693 EC50 = 630.96 nM T46185 C45ZNS 42596928 Ki = 5.754 nM T46185 C5DC7E 42598357 EC50 = 2511.89 nM T46185 CO6QB0 42598358 EC50 = 501.19 nM T46185 CDPA93 42598359 EC50 = 2511.89 nM T46185 CAM5P6 42598360 EC50 = 398.11 nM T46185 C58SRK 42598586 EC50 > 15848.93 nM T46185 CYL45Z 42598591 EC50 = 63.1 nM T46185 C6S2HI 42598828 EC50 = 794.33 nM T46185 C2GYA4 42598829 EC50 = 1258.93 nM T46185 C5CZ7P 42599068 EC50 = 630.96 nM T46185 C7O2ZV 42599070 EC50 = 100 nM T46185 C6BUZ5 42599071 EC50 = 794.33 nM T46185 CF23ZA 42853213 Ki = 794.33 nM T46185 CQJ5Z1 42853214 Ki = 199.53 nM T46185 CS40ML 44123747 IC50 > 10000 nM T46185 C8Z1XC 44134815 IC50 = 22 nM T46185 CMR7T1 44204999 EC50 > 25118.86 nM T46185 C3J2DY 44209166 EC50 = 14 nM T46185 CV1P7W 44213237 Ki = 20 nM T46185 CPW7K9 44232679 IC50 = 0.35 nM T46185 CU2T6F 44232680 IC50 = 0.73 nM T46185 CEQO63 44232682 IC50 = 0.44 nM T46185 CW1V2M 44232684 IC50 = 0.31 nM T46185 CDRG51 44232927 IC50 = 0.26 nM T46185 CVQB56 44232930 IC50 = 0.21 nM T46185 C4MK8P 44232931 IC50 = 0.23 nM T46185 CU6Q8I 44232952 Ki = 0.5012 nM T46185 C91ZIE 44232953 IC50 = 1553 nM T46185 C4OK7Y 44233172 IC50 = 0.36 nM T46185 C4Y3XC 44233174 IC50 = 2.24 nM T46185 CYC26A 44233176 IC50 = 0.27 nM T46185 C6WXJ9 44233187 IC50 = 458 nM T46185 CQM1T9 44233189 IC50 = 240 nM T46185 CAHP03 44233190 IC50 < 10 nM T46185 CA59KP 44233191 Ki = 3.981 nM T46185 C8LM6H 44233399 Ki = 0.08 nM T46185 CCK0D4 44233400 IC50 = 0.18 nM T46185 C3OY7U 44233402 IC50 = 0.17 nM T46185 CP1G4K 44233417 IC50 = 1273 nM T46185 CA7LB8 44233419 IC50 = 3478 nM T46185 C5Q3EJ 44233675 IC50 = 1195 nM T46185 CHK5U6 44233928 IC50 = 545 nM T46185 C9OG5Z 44234194 IC50 = 2119 nM T46185 CX21NW 44235638 IC50 = 79 nM T46185 C17PIF 44235871 IC50 = 1.14 nM T46185 CBU6A0 44236098 IC50 = 0.26 nM T46185 CK0JC2 44236099 IC50 = 0.54 nM T46185 CUD0K2 44236100 IC50 = 0.54 nM T46185 CG13KU 44236331 IC50 = 1.08 nM T46185 CH12JO 44236333 IC50 = 2.1 nM T46185 C73FXN 44236335 IC50 = 0.46 nM T46185 CR8WZ1 44236337 IC50 = 12 nM T46185 CA15LQ 44236339 IC50 = 0.38 nM T46185 CGR6J0 44251556 EC50 > 30000 nM T46185 C2K0VZ 44253016 EC50 = 79.43 nM T46185 CR2G0O 44265563 EC50 = 323.59 nM T46185 CT81XO 44265578 EC50 = 169.82 nM T46185 CG59FA 44267693 Ki = 22 nM T46185 CXS7F3 44267694 Ki = 250 nM T46185 CF6MX5 44267695 Ki = 1500 nM T46185 CHO0V6 44267696 Ki = 1 nM T46185 CBUN04 44267697 Ki = 256 nM T46185 CT70VP 44267699 Ki = 923 nM T46185 CSZ92K 44267703 Ki = 18 nM T46185 CJZA80 44267706 Ki = 2.7 nM T46185 CC3D2N 44267709 Ki = 48 nM T46185 CBYS94 44267712 Ki = 129 nM T46185 CV91YW 44267713 Ki = 108 nM T46185 CUM93G 44267714 Ki = 134 nM T46185 CKQH32 44267715 Ki = 254 nM T46185 C2BU1H 44267718 Ki = 11 nM T46185 C8TXY3 44267725 Ki = 20 nM T46185 CV17EJ 44267728 Ki = 14 nM T46185 CA4KC3 44267730 Ki = 4.3 nM T46185 C8P1LB 44267734 Ki = 40 nM T46185 CLDO45 44267740 Ki = 237 nM T46185 COQN60 44267744 Ki = 8.6 nM T46185 CN7QM3 44267747 Ki = 6.1 nM T46185 C7IP9N 44267748 Ki = 0.7 nM T46185 CY2D0W 44267749 Ki = 22 nM T46185 CQ4VW6 44267750 Ki = 256 nM T46185 CG95CQ 44267751 Ki = 26 nM T46185 CF4O7P 44267754 Ki = 134 nM T46185 CML7G8 44267758 Ki = 192 nM T46185 CB1KZ8 44267759 Ki = 12 nM T46185 C82HIW 44267762 Ki = 17 nM T46185 CNQP60 44267766 Ki = 104 nM T46185 C0D4EJ 44267772 Ki = 20 nM T46185 C1VG9X 44267782 Ki = 0.9 nM T46185 CF2A6M 44267796 Ki = 241 nM T46185 CM56OC 44267799 Ki = 260 nM T46185 C2LFH7 44274302 Ki = 12022.64 nM T46185 CZX4M3 44274317 Ki = 41686.94 nM T46185 C5L3FV 44274400 Ki = 29512.09 nM T46185 CF47ZS 44274417 Ki = 9120.11 nM T46185 CCK63Z 44274432 Ki = 14125.38 nM T46185 CZ1U0E 44274433 Ki = 15848.93 nM T46185 C3XP7C 44274441 Ki = 7413.1 nM T46185 CO1RL0 44274468 Ki = 15135.61 nM T46185 C9JX7D 44274469 Ki = 12589.25 nM T46185 CF36IC 44274477 Ki = 38904.51 nM T46185 CE20CZ 44275807 Ki = 933.25 nM T46185 CC2OD4 44278111 Ki > 10000 nM T46185 CRMA84 44278114 Ki > 10000 nM T46185 CF0Y4M 44278115 Ki > 10000 nM T46185 CFS16C 44285542 Ki > 20000 nM T46185 CSP92A 44285557 Ki = 15000 nM T46185 CR6D5Q 44285558 Ki > 25000 nM T46185 CXB29F 44285864 Ki > 20000 nM T46185 CRJ1X3 44295616 Ki = 104 nM T46185 CV7I2G 44295617 Ki = 1.9 nM T46185 CAVF41 44295618 Ki = 2.7 nM T46185 CH4Q3F 44295668 Ki = 78 nM T46185 CQ15FL 44295712 Ki = 5 nM T46185 CB6MT0 44295713 Ki = 122 nM T46185 CNF82K 44295763 Ki = 9 nM T46185 CA6UT5 44295787 Ki = 12 nM T46185 C02LYR 44295789 Ki = 15 nM T46185 C8XC2M 44295878 Ki = 106 nM T46185 C1YJ4B 44295888 Ki = 7 nM T46185 CA0Q7S 44295932 Ki = 1.6 nM T46185 C06FDI 44295953 Ki = 6 nM T46185 C4N6BC 44295954 Ki = 5 nM T46185 CQU2V5 44295965 Ki = 2.1 nM T46185 C3BDU0 44295977 Ki = 17 nM T46185 COL57Q 44296006 Ki = 9 nM T46185 CFW54U 44296007 Ki = 18 nM T46185 CI7G6Q 44296020 Ki = 27 nM T46185 C7IA6F 44296022 Ki = 40 nM T46185 CP7G2E 44296044 Ki = 1300 nM T46185 CU7YB3 44296053 Ki = 35 nM T46185 C5RI0Y 44296054 Ki = 2.4 nM T46185 CT31HC 44296096 Ki = 9 nM T46185 C1GX3I 44299477 Ki = 40 nM T46185 C9Z0LT 44299564 Ki = 851.14 nM T46185 CX28HR 44299589 Ki = 676.08 nM T46185 CPL36O 44299599 Ki = 1174.9 nM T46185 CFN95A 44299616 Ki = 1737.8 nM T46185 CE4L1V 44299635 Ki = 1148.15 nM T46185 C9TWN3 44302727 IC50 = 3002.9 nM T46185 C5S8UL 44302728 IC50 = 9341.4 nM T46185 CQ4B5T 44302741 IC50 = 1905.1 nM T46185 C0AZF5 44302755 IC50 = 7703.7 nM T46185 CR5T1J 44302775 IC50 = 2565 nM T46185 CY8PD1 44302776 IC50 = 9524.7 nM T46185 C7GY5J 44302788 IC50 = 13138 nM T46185 CAV72D 44302793 IC50 = 14677.7 nM T46185 CV9QM6 44302813 IC50 = 2680.7 nM T46185 C43QTF 44302833 IC50 < 1000 nM T46185 CF74EQ 44302834 IC50 = 1646 nM T46185 C6J3EY 44302879 IC50 = 4662.4 nM T46185 CIU20B 44302900 IC50 = 2643 nM T46185 CGNA91 44302901 IC50 = 1151.5 nM T46185 CQPV04 44303017 EC50 = 1210 nM T46185 CY47SI 44303018 EC50 = 2280 nM T46185 C6H2ZT 44303019 EC50 = 791 nM T46185 C6BMW2 44303286 EC50 = 779 nM T46185 C3L8RU 44303293 EC50 = 528 nM T46185 C0SLC4 44303294 EC50 = 763 nM T46185 C7X1GV 44303314 EC50 = 904 nM T46185 C85QFH 44303323 EC50 = 83 nM T46185 C7J1HZ 44303327 EC50 = 853 nM T46185 CD9A5N 44303396 EC50 = 80 nM T46185 CW6O3V 44303397 EC50 = 673 nM T46185 C5VJK4 44303408 EC50 = 1480 nM T46185 C1RGS9 44304818 Ki = 480 nM T46185 C03MFZ 44308733 Ki = 210 nM T46185 CT3V7Z 44308746 Ki = 640 nM T46185 C0Z3JQ 44308798 Ki = 36000 nM T46185 CN9M6A 44308799 Ki = 15000 nM T46185 C38WIK 44308809 Ki = 6800 nM T46185 CF06ON 44308818 Ki = 2900 nM T46185 C90FZB 44308831 Ki = 5400 nM T46185 CK14IH 44308832 Ki = 55 nM T46185 COE23J 44308861 Ki = 28 nM T46185 CMX10C 44308899 Ki = 41 nM T46185 CN5G8U 44308900 Ki = 820 nM T46185 CLJ71S 44308910 Ki = 1200 nM T46185 C3L7HC 44308912 Ki = 130 nM T46185 CP0G8R 44308913 Ki = 300 nM T46185 CY6TU4 44309089 Ki = 2200 nM T46185 CMAC70 44309090 Ki = 3900 nM T46185 CND98T 44309107 Ki = 5300 nM T46185 CEFY94 44309108 Ki = 15000 nM T46185 C61LZX 44309135 Ki = 4200 nM T46185 CY8D9F 44309151 Ki = 2800 nM T46185 CD7QT6 44309153 Ki = 760 nM T46185 C7CQ3N 44309208 Ki = 1100 nM T46185 C3B0IJ 44309209 Ki = 1000 nM T46185 CIG89A 44309231 Ki = 300 nM T46185 CSW73I 44311704 Ki = 2.198 nM T46185 C2R3SX 44311716 Ki = 1.449 nM T46185 CJ9C3I 44311717 Ki = 0.3597 nM T46185 C7QD0Y 44311718 Ki = 0.38 nM T46185 CH7IJ2 44311760 Ki = 0.38 nM T46185 CGY95E 44311761 Ki = 3.8 nM T46185 CT41MZ 44311762 Ki = 1.14 nM T46185 CT6Y9V 44311771 Ki = 0.2897 nM T46185 CJ3F7Y 44311784 Ki = 0.3499 nM T46185 CO28DW 44311785 Ki = 0.59 nM T46185 CI2LP0 44311786 Ki = 0.99 nM T46185 CV52TA 44311823 Ki = 0.4498 nM T46185 CQ51WZ 44311835 Ki = 2.99 nM T46185 CT8U1D 44311987 Ki = 0.46 nM T46185 CSA8M2 44312007 Ki = 0.2999 nM T46185 C4ENG6 44312024 Ki = 0.41 nM T46185 CBE37N 44312066 Ki = 17 nM T46185 C7W3FI 44312081 Ki = 37 nM T46185 C6OP9A 44312083 Ki = 0.8 nM T46185 COX3S1 44312132 Ki = 4600 nM T46185 C89QFR 44312152 Ki = 26 nM T46185 CZ65YU 44312450 Ki = 0.6 nM T46185 C6YGO9 44312451 Ki = 0.6 nM T46185 CZ84YU 44312455 Ki = 36 nM T46185 CWN9H1 44312460 Ki = 34 nM T46185 CL6M1O 44312464 Ki = 33 nM T46185 CP4S2D 44312468 Ki = 135 nM T46185 CM0Z7K 44313166 Ki = 1189 nM T46185 CU9FV1 44313489 Ki = 500 nM T46185 CC5W6M 44313626 Ki = 74 nM T46185 C04VNU 44313630 Ki = 22 nM T46185 C71NXG 44313631 Ki > 10000 nM T46185 CO0J3B 44314328 Ki = 0.29 nM T46185 C8O4SV 44314329 Ki = 0.99 nM T46185 C1CAH2 44314347 Ki = 0.14 nM T46185 C4C8LW 44314554 Ki = 33.3 nM T46185 C7BQ0K 44314564 Ki = 0.23 nM T46185 C8X7PS 44314697 Ki = 0.2 nM T46185 CHU4N2 44314698 Ki = 0.81 nM T46185 C3ZG7W 44314699 Ki = 1.2 nM T46185 CIM4P3 44314713 Ki = 1.4 nM T46185 CVX13Q 44318736 Ki = 310 nM T46185 CT58BQ 44318766 Ki = 3600 nM T46185 CLDG78 44318781 Ki = 3981.07 nM T46185 CAH58Q 44318782 Ki = 19.95 nM T46185 CR2T3J 44318817 Ki = 1200 nM T46185 C89JNT 44318928 Ki = 125.89 nM T46185 CL0HY5 44318929 Ki = 820 nM T46185 C01CVA 44318930 Ki = 730 nM T46185 C9Q6ET 44318969 Ki = 630.96 nM T46185 CZOA25 44319006 Ki = 316.23 nM T46185 CM0VD2 44319008 Ki = 398.11 nM T46185 CP9WF7 44319009 Ki = 19.95 nM T46185 C46OXB 44319010 Ki = 251.19 nM T46185 CT07JE 44319016 Ki = 630.96 nM T46185 CZ96OC 44319017 Ki = 630.96 nM T46185 C0C2XL 44319043 Ki = 50.12 nM T46185 C9SDP3 44319071 Ki = 7.943 nM T46185 C7R9DO 44319339 Ki = 79.43 nM T46185 C93POZ 44319342 Ki = 25.12 nM T46185 CM9RX2 44324655 Ki = 0.72 nM T46185 CKYH35 44324848 Ki = 14.3 nM T46185 CDQ7M2 44324891 Ki = 1.82 nM T46185 C8QT4C 44324892 Ki = 0.03 nM T46185 CD6E8X 44325003 Ki = 9.09 nM T46185 C6M5XU 44325013 Ki = 5.07 nM T46185 CU1K3L 44325017 Ki = 0.82 nM T46185 CFE8L2 44325018 Ki = 0.031 nM T46185 CF03PV 44325034 Ki = 1.22 nM T46185 C7GQI9 44325047 Ki = 0.823 nM T46185 CYG46U 44325048 Ki = 0.16 nM T46185 CW2K7D 44325051 Ki = 34.8 nM T46185 CUB76V 44325052 Ki = 1.02 nM T46185 CT3GJ1 44325080 Ki = 12.1 nM T46185 CGSU92 44326538 Ki = 243 nM T46185 CSE35C 44328347 Ki = 2400 nM T46185 CM6D4U 44328348 Ki > 5000 nM T46185 CX4M2I 44328356 Ki > 8000 nM T46185 C8O4PB 44328540 Ki = 2200 nM T46185 CTX68J 44328560 Ki >> 200 nM T46185 CP5W3M 44328561 Ki = 1700 nM T46185 CO18HJ 44329977 EC50 = 11 nM T46185 CDC01L 44330073 EC50 = 139 nM T46185 CYC95E 44330074 EC50 > 10000 nM T46185 CL5EU8 44330080 EC50 = 227 nM T46185 CBTX60 44330081 EC50 = 9 nM T46185 CPGN89 44337326 Ki = 1.3 nM T46185 CD9ZS8 44342270 IC50 = 1570 nM T46185 CSK4B0 44346542 IC50 = 2734.2 nM T46185 CU2X1V 44356367 IC50 = 18000 nM T46185 CXJ4G7 44364174 Ki = 2300 nM T46185 CAM9P4 44378597 Ki = 1.3 nM T46185 CE6YC8 44378598 Ki = 3 nM T46185 C7SM6N 44378599 Ki = 4.7 nM T46185 CRF7X6 44378600 Ki = 442 nM T46185 CJ7T6W 44378601 Ki = 0.2 nM T46185 CYGD60 44378689 Ki = 0.8 nM T46185 CI9R0S 44378753 Ki = 16 nM T46185 C30AKW 44378762 Ki = 0.03 nM T46185 CJ2VA1 44378763 Ki = 1.8 nM T46185 CQ1C7W 44378764 Ki = 0.4 nM T46185 C2L7CS 44378765 Ki = 2.5 nM T46185 C6T4DY 44378769 Ki = 53 nM T46185 CCPB86 44378810 Ki = 0.3 nM T46185 C4N2RC 44378811 Ki = 0.04 nM T46185 C1CV2H 44378842 Ki = 0.2 nM T46185 CW6CG2 44378845 Ki = 0.03 nM T46185 CYC1A7 44378846 Ki = 0.14 nM T46185 CZ61WT 44378862 Ki = 2.6 nM T46185 CFU79I 44378875 Ki = 0.1 nM T46185 C3U6ZK 44378876 Ki = 0.3 nM T46185 CX9GP3 44378888 Ki = 77 nM T46185 C3FT5L 44378951 Ki = 1 nM T46185 CZXK89 44378952 Ki = 0.3 nM T46185 C28RUJ 44378958 Ki = 0.8 nM T46185 CEWZ65 44378982 Ki = 4.4 nM T46185 C1SD8K 44379021 Ki = 0.1 nM T46185 C4R3IU 44379026 Ki = 0.16 nM T46185 C1S9IB 44379040 Ki = 0.5 nM T46185 C6S5QA 44379050 Ki = 0.2 nM T46185 C17PJS 44379051 Ki = 0.1 nM T46185 CX6GA3 44379052 Ki = 1.3 nM T46185 C32DXF 44379055 Ki = 0.6 nM T46185 C3VT2M 44379080 Ki = 46.9 nM T46185 CU68GE 44379281 Ki = 37.1 nM T46185 CUA24S 44379508 Ki = 111 nM T46185 CZ4X3O 44382125 Ki = 138.8 nM T46185 C6EOV3 44382247 Ki = 34.7 nM T46185 C9Z0AB 44382606 Ki = 0.5 nM T46185 CNW6X2 44382652 Ki = 14 nM T46185 CUF3E0 44382699 Ki = 3.2 nM T46185 CMFC59 44382739 Ki = 6 nM T46185 CQ7P3Y 44382840 Ki = 376 nM T46185 CCYU52 44382841 Ki = 189 nM T46185 CW2J6Y 44382858 Ki = 352 nM T46185 C7VOM3 44382864 Ki > 280 nM T46185 CKC6L3 44382865 Ki = 224 nM T46185 C8OZ2J 44382880 Ki = 570 nM T46185 C3TX9A 44382974 Ki = 520 nM T46185 C5JHQ8 44383064 Ki = 184 nM T46185 C26DNS 44383065 Ki = 26 nM T46185 CO3UJ2 44383238 Ki = 13 nM T46185 C7H6ZY 44383305 Ki = 59.5 nM T46185 CDR8O5 44383342 Ki = 1.6 nM T46185 C61QNW 44383352 Ki = 650 nM T46185 C0G2RO 44383373 Ki = 595 nM T46185 CEZ56X 44383415 Ki = 17.9 nM T46185 CXG5Q3 44383489 Ki = 485 nM T46185 C1BP8Z 44383490 Ki > 500 nM T46185 C9T1BR 44383492 Ki > 500 nM T46185 CG90DX 44383554 Ki = 312 nM T46185 CA8T0K 44383595 Ki = 209 nM T46185 CDA8W1 44383613 Ki > 500 nM T46185 C5X3RM 44383653 Ki = 4.3 nM T46185 CZ8E1C 44383766 Ki > 42 nM T46185 CY6B5S 44384258 Ki = 275 nM T46185 C36YBR 44384326 Ki = 283 nM T46185 CIDW56 44384327 Ki = 148 nM T46185 C7YTV9 44385809 Ki = 270 nM T46185 CHD9O7 44386115 Ki = 17 nM T46185 CG2VT0 44392899 Ki > 1400 nM T46185 CFY5B7 44392905 Ki = 180 nM T46185 CIW3F6 44392933 Ki = 16 nM T46185 C1GB6S 44392936 Ki > 1400 nM T46185 CCX9A6 44392956 Ki > 1400 nM T46185 C2H4QG 44392960 Ki = 43 nM T46185 C0HP4R 44392966 Ki = 12.2 nM T46185 C3MKY5 44392967 Ki = 449 nM T46185 CPVS57 44392974 Ki = 68 nM T46185 CD5PS0 44392978 Ki > 1400 nM T46185 CS8F0W 44392983 Ki = 571 nM T46185 C1B4QL 44403095 Ki > 10000 nM T46185 C1YL7Z 44403098 Ki > 10000 nM T46185 CFV98A 44403101 Ki > 10000 nM T46185 C6OY9S 44403102 Ki > 10000 nM T46185 CH4SX6 44403105 Ki > 10000 nM T46185 C12FIH 44403106 Ki > 10000 nM T46185 C4LKC1 44404394 Ki > 10000 nM T46185 C3EJ4G 44404396 Ki > 10000 nM T46185 CT8S1N 44406268 Ki = 20 nM T46185 C43QUG 44406316 Ki = 40 nM T46185 C6B1HT 44406321 Ki = 126 nM T46185 CO14PG 44406342 Ki = 3161 nM T46185 CPYG54 44406346 Ki = 251 nM T46185 CX7SG3 44406387 Ki = 501 nM T46185 C3G6PR 44406395 Ki = 50 nM T46185 C3UAN2 44406406 Ki = 50 nM T46185 C6I3KL 44406451 Ki = 631 nM T46185 CX6L1E 44406476 Ki = 316 nM T46185 CMR10G 44406480 Ki = 79 nM T46185 C4SC6T 44406481 Ki = 1.3 nM T46185 C16NYM 44406520 Ki = 50 nM T46185 CVL24Q 44406521 Ki = 5 nM T46185 C3ZV2I 44406527 Ki = 100 nM T46185 CQCH24 44406572 Ki = 251 nM T46185 CRMB45 44406573 Ki = 2 nM T46185 CH5D2N 44406597 Ki = 3.2 nM T46185 C0A1PB 44406598 Ki = 13 nM T46185 CY0DB3 44406662 Ki = 4 nM T46185 CZM93T 44406686 Ki = 3.2 nM T46185 CZX87U 44406689 Ki = 40 nM T46185 CP0J2E 44406690 Ki = 2 nM T46185 C6GLV1 44408714 Ki = 3235.94 nM T46185 CG9Y5H 44408892 EC50 = 446.68 nM T46185 COX8D7 44408895 EC50 = 229.09 nM T46185 CR6CE1 44408940 EC50 = 109.65 nM T46185 C4QTI3 44415886 Ki = 1500 nM T46185 CC9AV3 44418764 Ki = 39.81 nM T46185 CV6UQ3 44419370 Ki > 100000 nM T46185 C84KBW 44420791 Ki = 498 nM T46185 C2P7XQ 44420794 Ki = 5.4 nM T46185 CS9XH3 44420821 Ki = 65 nM T46185 C2N5LX 44422691 Ki = 2089.3 nM T46185 CIRB78 44422696 Ki = 5248.07 nM T46185 CHT24X 44422698 Ki = 6918.31 nM T46185 CDE8A1 44428745 Ki = 6.026 nM T46185 CRN6M1 44431367 Ki = 90 nM T46185 CQD71K 44431369 Ki = 48 nM T46185 CAE86V 44431370 Ki = 49 nM T46185 C92HNF 44431372 Ki = 44 nM T46185 CI36TZ 44431375 Ki = 49 nM T46185 CZ12VG 44431376 Ki = 41 nM T46185 CS0H4C 44431380 Ki = 12 nM T46185 C5FJR6 44431381 Ki = 2.4 nM T46185 CG0BM9 44431382 Ki = 6.2 nM T46185 CW60PY 44431383 Ki = 2 nM T46185 C0JL9K 44431384 Ki = 0.66 nM T46185 C3S0AU 44431386 Ki = 8.8 nM T46185 C0T5AL 44431387 Ki = 7.2 nM T46185 C15WZI 44431388 Ki = 12 nM T46185 C29VWS 44431389 Ki = 1.9 nM T46185 C1LJ6G 44431391 Ki = 5.1 nM T46185 CLA76R 44431393 Ki = 0.12 nM T46185 CG45PO 44437242 Ki = 50 nM T46185 C6I2JO 44437248 Ki = 2041 nM T46185 CZI05O 44437258 Ki > 10000 nM T46185 C2DAH1 44437265 Ki > 10000 nM T46185 C2EFY1 44437274 Ki > 10000 nM T46185 CXD1P2 44437278 Ki > 10000 nM T46185 C3E5FV 44437285 Ki > 10000 nM T46185 C7VP1Y 44437297 Ki = 219 nM T46185 C5GT7C 44437302 Ki = 4099 nM T46185 C37QFT 44437307 Ki = 474 nM T46185 C36LXN 44446840 Ki = 4897.79 nM T46185 CVT7J2 44449463 Ki = 31.62 nM T46185 CR4ZT2 44450620 Ki = 5248.07 nM T46185 C5H7OQ 44450621 Ki = 3548.13 nM T46185 CZ50IM 44450622 Ki = 1412.54 nM T46185 CS5CD3 44450624 Ki = 676.08 nM T46185 CFN4B5 44450637 Ki = 1698.24 nM T46185 C12XGE 44456400 Ki > 10000 nM T46185 C4DL5C 44469677 IC50 > 10000 nM T46185 CVA67X 44568347 Ki = 220 nM T46185 CY9C2A 44571572 Ki > 100000 nM T46185 CM0D1J 44575653 IC50 = 6 nM T46185 CN68YI 44578707 Ki = 645.65 nM T46185 CHUN40 44578928 EC50 > 50000 nM T46185 CZYP06 44578975 EC50 > 50000 nM T46185 CCIT12 44578976 EC50 > 50000 nM T46185 CW53ZF 44578977 EC50 > 50000 nM T46185 CYHM34 44578978 EC50 > 50000 nM T46185 CGF7A4 44579375 EC50 > 50000 nM T46185 C1OCB6 44579416 EC50 > 50000 nM T46185 CARW17 44579417 EC50 > 50000 nM T46185 C2DFV7 44579418 EC50 > 50000 nM T46185 CTC8H6 44579419 EC50 > 50000 nM T46185 CYR0O3 44579457 EC50 > 50000 nM T46185 CF1EA4 44579458 EC50 > 50000 nM T46185 C6HMP4 44589495 IC50 = 100 nM T46185 C9U3KY 44589496 IC50 = 79.43 nM T46185 CXL82E 44589497 IC50 = 1258.93 nM T46185 CLGW57 44589498 IC50 = 398.11 nM T46185 C1KY5I 44589499 IC50 > 3162.28 nM T46185 C0N4QF 44589529 IC50 > 3162.28 nM T46185 CQ4Y8O 44589531 EC50 > 30000 nM T46185 COE0T7 44589569 IC50 > 3162.28 nM T46185 CE4FX5 44589570 IC50 = 1584.89 nM T46185 C9J2RO 44589571 IC50 = 1584.89 nM T46185 CKY4F8 44589572 IC50 > 3162.28 nM T46185 CX19BO 44589573 IC50 > 3162.28 nM T46185 C10LXB 44589574 IC50 > 3162.28 nM T46185 CUD4M8 44589575 IC50 > 3162.28 nM T46185 CL40CM 44589593 EC50 > 30000 nM T46185 CKS5V4 44589594 EC50 > 30000 nM T46185 CXB30W 44589595 EC50 > 30000 nM T46185 CM5LJ8 44589596 EC50 > 30000 nM T46185 CPXE19 44589643 EC50 > 30000 nM T46185 C8AJO6 44589644 EC50 > 30000 nM T46185 CFS1A4 44589645 EC50 > 30000 nM T46185 C71EHI 44589646 EC50 > 30000 nM T46185 CQB5A9 44589681 EC50 = 11.9 nM T46185 CE06LX 44589984 IC50 = 158.49 nM T46185 C6LC7V 44590033 IC50 = 251.19 nM T46185 CL57OY 44590034 IC50 = 316.23 nM T46185 CO3GX2 44590035 IC50 = 158.49 nM T46185 CT58OX 44590036 IC50 = 199.53 nM T46185 C2H9IW 44590122 IC50 = 100 nM T46185 CJ2M0R 44590123 IC50 = 125.89 nM T46185 C5JVF6 44590124 IC50 = 630.96 nM T46185 C3G5LY 44590125 IC50 = 199.53 nM T46185 CF4DI1 44590166 IC50 = 2511.89 nM T46185 CYC47W 44590167 IC50 = 100 nM T46185 CH61KJ 44590182 IC50 = 316.23 nM T46185 CUA62X 44593616 Ki = 39.81 nM T46185 CN9ID8 44593617 Ki = 218.78 nM T46185 CDM56I 44593618 Ki = 4.169 nM T46185 CU63PQ 44593619 Ki = 64.57 nM T46185 CL8D2S 44593620 Ki = 38.02 nM T46185 CI97KQ 44593621 Ki = 302 nM T46185 CNZ1U7 44593651 IC50 < 1 nM T46185 CL5O8E 44602489 EC50 > 30000 nM T46185 CH2Z3O 44610056 Ki = 0.14 nM T46185 CVZ6Y1 44627739 Ki = 29.51 nM T46185 CE6A9F 44627740 Ki = 6.761 nM T46185 C6EU7P 44627741 Ki = 64.57 nM T46185 CW40TR 44627742 Ki = 141.25 nM T46185 C5GIU6 44627743 Ki = 31.62 nM T46185 CK9DO1 44627745 Ki = 10.23 nM T46185 CJ8S1L 44627747 Ki = 13.49 nM T46185 C5LY8C 44627851 Ki = 17.38 nM T46185 CC4A3X 44627853 Ki = 4.571 nM T46185 CH4N5J 44627854 Ki = 60.26 nM T46185 CO8C6D 44627855 Ki = 363.08 nM T46185 COL8E1 44627856 Ki = 3235.94 nM T46185 C6WS7M 44627857 Ki = 2.344 nM T46185 C43BJY 44627859 Ki = 19.95 nM T46185 CW0X6A 44627955 Ki = 87.1 nM T46185 CXNF31 44627957 Ki = 758.58 nM T46185 C4LOY2 45115589 Ki < 1000 nM T46185 C9U0VH 45259185 Ki = 69.18 nM T46185 CNC1R2 45259186 Ki = 41.69 nM T46185 CP2CZ7 45259187 Ki = 85.11 nM T46185 CW14TS 45259188 Ki = 17.78 nM T46185 CO8W1X 45259189 Ki = 21.38 nM T46185 CF16YZ 45259190 Ki = 57.54 nM T46185 C1K0ZH 45259193 Ki = 3.162 nM T46185 C7L1CU 45266348 Ki = 74.13 nM T46185 CP3J5W 45266385 Ki = 77624.71 nM T46185 CK8N4L 45266386 Ki = 9332.54 nM T46185 CJQ8C6 45266387 IC50 = 5.012 nM T46185 C2IV6N 45266389 IC50 = 3.981 nM T46185 C7WBU9 45266390 IC50 = 10 nM T46185 C5J2TE 45266397 IC50 = 39.81 nM T46185 C0O9TA 45266401 IC50 = 12.59 nM T46185 C5P1NR 45266404 IC50 = 100 nM T46185 CJ9W5C 45266406 IC50 = 39.81 nM T46185 CH74XR 45266408 IC50 = 3.981 nM T46185 CGH8T0 45266411 IC50 = 50.12 nM T46185 C73TVO 45266437 IC50 = 10 nM T46185 C5PTZ9 45266459 IC50 = 5.012 nM T46185 C0D4LK 45266462 IC50 = 15.85 nM T46185 CUK8N1 45266464 IC50 = 12.59 nM T46185 CRI98L 45266467 IC50 = 39.81 nM T46185 C0AV6F 45266469 IC50 = 2.512 nM T46185 CZA73U 45266470 IC50 = 2.512 nM T46185 C0FHW1 45266476 IC50 = 10 nM T46185 CZ23VF 45266478 IC50 = 6.31 nM T46185 CK6X3B 45786849 EC50 = 13000 nM T46185 CL0M1G 46174144 Ki = 0.1585 nM T46185 CU4V5R 46227410 Ki = 17378.01 nM T46185 CWQ1L9 46227412 Ki = 13803.84 nM T46185 CX2E6A 46227414 Ki = 16595.87 nM T46185 C0Z4RD 46227416 Ki = 89125.09 nM T46185 CK2R5G 46227454 Ki = 19952.62 nM T46185 C8OZI6 46227456 Ki = 18197.01 nM T46185 CB45NM 46227458 Ki = 95499.26 nM T46185 C1J0IF 46227460 Ki = 60255.96 nM T46185 CQ4DI6 46227480 Ki = 72443.6 nM T46185 CHKL80 46227482 Ki = 27542.29 nM T46185 CVP7T6 46227484 Ki = 33884.42 nM T46185 CC6RH5 46227486 Ki = 46773.51 nM T46185 CSQ0V3 46227554 Ki = 11220.18 nM T46185 C1Q0MH 46830362 IC50 = 2700 nM T46185 CH3ID7 46830363 IC50 > 10000 nM T46185 CH83EL 46854806 EC50 = 0.28 nM T46185 CI6SN1 46855274 Ki = 100 nM T46185 C01YTE 46871665 IC50 = 1995.26 nM T46185 CUY51M 46871666 IC50 = 3981.07 nM T46185 CYLZ50 46871844 IC50 = 199.53 nM T46185 CNA6C1 46878253 EC50 = 11.22 nM T46185 CY7P0I 46878255 EC50 = 8.128 nM T46185 CCZ5I8 46883796 IC50 > 10000 nM T46185 CVCF68 46883843 IC50 > 10000 nM T46185 CW70YU 46890977 IC50 = 398.11 nM T46185 CJ74AZ 46891076 IC50 = 1258.93 nM T46185 CTSZ49 46891179 IC50 = 2511.89 nM T46185 COT8S4 46891375 EC50 > 10000 nM T46185 CW1YX7 46891488 IC50 = 7943.28 nM T46185 CB1Z5A 46905390 IC50 = 1637.8 nM T46185 C67XQI 46945663 EC50 > 30000 nM T46185 C7IAW9 49663949 IC50 < 1500 nM T46185 CD39WZ 49665121 IC50 = 930 nM T46185 C2LZJ0 49783209 Ki = 433 nM T46185 C57SMG 49783415 Ki > 10000 nM T46185 C0TG6I 49783419 Ki > 10000 nM T46185 C2TAI1 49797319 Ki > 10000 nM T46185 C20SCO 49797320 Ki > 10000 nM T46185 C29QSB 49797322 Ki = 40 nM T46185 CHS34N 49797323 Ki > 10000 nM T46185 C9V5OK 49797324 Ki > 10000 nM T46185 CT4QU7 49797325 Ki = 876 nM T46185 C1WG5X 49797326 Ki > 10000 nM T46185 C13SKB 49797327 Ki > 10000 nM T46185 CLB8A4 49797328 Ki > 10000 nM T46185 CGB63L 49799920 EC50 = 1075 nM T46185 CPI6N0 49853777 IC50 > 100000 nM T46185 C94GDK 49853778 IC50 > 100000 nM T46185 CHV3U8 49853881 IC50 > 100000 nM T46185 CTBY97 49853883 IC50 > 100000 nM T46185 CQP63D 49853884 IC50 = 93000 nM T46185 CY8M9A 49853885 IC50 > 100000 nM T46185 CN0JU9 49853987 IC50 > 100000 nM T46185 C8DVX6 49855131 IC50 > 100000 nM T46185 C2RY0J 50878551 Ki > 10000 nM T46185 C1W6TV 50898777 Ki = 2511.89 nM T46185 CXMZ73 50898778 Ki > 10000 nM T46185 C3BZ7G 50925541 IC50 = 3.162 nM T46185 C7NGS9 50925542 IC50 = 1.259 nM T46185 CHG0K5 50925543 IC50 = 3.162 nM T46185 CE4KP1 51050257 Ki > 10000 nM T46185 CM47HJ 52176747 IC50 = 1200 nM T46185 C80EHA 52941205 Ki = 10.38 nM T46185 CT16AY 52942401 IC50 = 25.12 nM T46185 CY6UC5 52942402 IC50 = 10 nM T46185 CLXF87 52942447 IC50 > 1000 nM T46185 CYQF74 52942458 IC50 = 3.981 nM T46185 CM3IV9 52942497 IC50 = 79.43 nM T46185 C1G7HW 52942610 IC50 = 125.89 nM T46185 CZ3X0R 52942628 IC50 = 25.12 nM T46185 CXT1M9 52943696 IC50 = 6.31 nM T46185 CZ78UX 52943721 IC50 = 15.85 nM T46185 C5O4MA 52943879 IC50 = 50.12 nM T46185 C5UN3Y 52943921 IC50 = 125.89 nM T46185 CFLA17 52944764 IC50 > 1000 nM T46185 CE04VX 52945165 IC50 = 79.43 nM T46185 C7YT1B 52945255 IC50 = 251.19 nM T46185 CBTM43 52945272 IC50 = 15.85 nM T46185 CW49GK 52946068 IC50 = 794.33 nM T46185 C6YBT4 52946249 IC50 = 19.95 nM T46185 CJ85YX 52946359 IC50 = 39.81 nM T46185 CZT9U3 52947254 IC50 = 31.62 nM T46185 COW8Z9 52947320 IC50 = 2.512 nM T46185 C7QNY8 52947416 IC50 = 794.33 nM T46185 CV81IX 52947552 IC50 = 125.89 nM T46185 CC4A1H 52947553 IC50 = 63.1 nM T46185 CF08DE 52948443 IC50 = 12.59 nM T46185 CBQ7X1 52949760 IC50 > 1000 nM T46185 CN91QX 52949883 IC50 = 79.43 nM T46185 CN0U6H 52949961 IC50 = 31.62 nM T46185 C2LEQ0 52950036 IC50 = 50.12 nM T46185 C6KU3Z 53303986 IC50 > 10000 nM T46185 CR4W9L 53324553 Ki = 2287 nM T46185 C28QUB 53373577 Ki < 38018.94 nM T46185 CS1OI7 53382523 EC50 > 30000 nM T46185 CWR16G 53382542 EC50 = 550 nM T46185 C7YP3A 53385782 EC50 = 1800 nM T46185 CPGC12 53385783 EC50 > 10000 nM T46185 CC8Q1D 53390181 Ki = 870.96 nM T46185 CV0P1K 53390538 Ki = 870.96 nM T46185 CZ0WI6 53391301 Ki = 1621.81 nM T46185 C6A7VE 53414666 Ki = 11000 nM T46185 C6D3OU 54580864 IC50 = 14.4 nM T46185 CM9KH3 54581928 IC50 = 120.8 nM T46185 C1ZMV9 54582844 IC50 = 28 nM T46185 CMRC75 54583839 IC50 = 349.3 nM T46185 CZ82MJ 54583840 IC50 = 45.8 nM T46185 C01VQF 54584800 IC50 = 88.9 nM T46185 CHP9F8 54585742 IC50 = 2779 nM T46185 CO5H6T 54585743 IC50 = 26.8 nM T46185 CB5IF2 54586723 IC50 = 1364.9 nM T46185 CKTW24 54586742 IC50 = 33.1 nM T46185 CWXP12 54586744 IC50 = 29.8 nM T46185 CK01PH 54757332 Ki = 15 nM T46185 C8WHT5 56593934 Ki = 10000 nM T46185 CA9T3J 56667295 Ki = 0.68 nM T46185 CU0NE5 56672197 Ki = 3542 nM T46185 CB0P9N 56944383 Ki > 1000 nM T46185 C1TC7Q 56963799 Ki = 681 nM T46185 C3WC7Z 56965018 Ki = 16.6 nM T46185 CP53TW 57088082 EC50 = 29 nM T46185 CL8C4R 57230548 EC50 = 2253 nM T46185 CUP4Y0 57326139 Ki = 6309.57 nM T46185 C1G9XY 57326141 Ki = 18197.01 nM T46185 CG3YS9 57326143 Ki = 6456.54 nM T46185 CCYU25 57326145 Ki = 39810.72 nM T46185 CS86GL 57326232 Ki = 33.11 nM T46185 C3AF0Z 57326234 Ki = 2.818 nM T46185 CLSW35 57326236 Ki = 28183.83 nM T46185 CL3R5D 57326238 Ki = 79432.82 nM T46185 C4G1LB 57326325 Ki = 95.5 nM T46185 C6CB9J 57326326 Ki = 9.772 nM T46185 C5OJP0 57391102 EC50 > 30000 nM T46185 C17GMJ 57393065 IC50 > 30000 nM T46185 C6HBG0 57396813 IC50 = 7900 nM T46185 CQ5BG6 57525860 EC50 > 30000 nM T46185 C9TMZ3 57558000 Ki > 100000 nM T46185 C54DIC 58438451 Ki = 21877.62 nM T46185 C9UK7P 58438475 Ki = 14125.38 nM T46185 CBCA81 58438487 Ki < 67608.3 nM T46185 CA14SG 58653718 Ki > 100000 nM T46185 C2XDJ0 58975257 IC50 = 5345 nM T46185 CRV9X7 59654579 EC50 = 71.8 nM T46185 C6C7EJ 60138185 Ki = 75.86 nM T46185 C8WGS2 60138186 Ki = 61.66 nM T46185 CAZ9B3 62705488 IC50 > 10000 nM T46185 C9F4JW 62705832 IC50 > 10000 nM T46185 CA5FP7 66561966 Ki = 4738 nM T46185 C3XL7O 66561967 Ki = 696 nM T46185 C9A8WH 66875589 Ki = 6.31 nM T46185 C4UP0J 67405379 Ki < 56234.13 nM T46185 CU32ZC 67407161 Ki = 28183.83 nM T46185 C3GSR6 67407808 Ki < 67608.3 nM T46185 CWY79V 67408128 Ki < 54954.09 nM T46185 CB06GE 67547652 IC50 = 285.9 nM T46185 CDH6V7 67547661 IC50 = 804.2 nM T46185 CE91TN 67547949 IC50 = 136.6 nM T46185 CMA5W7 67548135 IC50 = 0.9 nM T46185 C8OC2K 67548543 IC50 = 140.2 nM T46185 CD41JS 67548925 IC50 = 0.6 nM T46185 C8MU9E 67549179 IC50 = 101.1 nM T46185 CCB1T5 68764898 Ki = 4010 nM T46185 CTW10U 69058945 Ki = 3.981 nM T46185 C6TI9M 69444105 IC50 = 38.2 nM T46185 CF8DC9 70681307 Ki = 4.467 nM T46185 CKSP64 70682037 Ki = 269.15 nM T46185 CXT67P 70683405 Ki = 5.37 nM T46185 CN98LU 70685504 Ki = 3.467 nM T46185 CT41UM 70687661 Ki = 3.981 nM T46185 C5AR1G 70693619 Ki = 45000 nM T46185 CJLS94 71449148 Ki = 7.67 nM T46185 C9VZ8J 71450550 Ki = 666 nM T46185 C4M1WQ 71450615 IC50 = 311.2 nM T46185 C29VNS 71450616 IC50 = 13.1 nM T46185 CDN70A 71450617 IC50 = 336.8 nM T46185 C8HR1L 71450662 IC50 = 410.6 nM T46185 CY3M8B 71451570 IC50 > 1500 nM T46185 C4NDR3 71452382 Ki = 216 nM T46185 CYK20Z 71452384 Ki = 872 nM T46185 CDTW09 71452387 Ki = 1295 nM T46185 C54WNK 71452454 IC50 = 427 nM T46185 CPO41L 71452455 IC50 = 191 nM T46185 CYF3R2 71452456 IC50 = 327.8 nM T46185 C5WK8L 71452756 Ki = 0.03 nM T46185 CK81FI 71452793 Ki = 10.8 nM T46185 CG4ZX5 71454212 IC50 = 87.6 nM T46185 CSJ16R 71454213 IC50 = 41.2 nM T46185 CRMC04 71454214 IC50 = 860.2 nM T46185 CZS9G3 71454215 IC50 = 181.2 nM T46185 CR41KC 71454216 IC50 < 5 nM T46185 C5OBD0 71454217 IC50 = 555.9 nM T46185 CX26PA 71454562 Ki = 7.14 nM T46185 CX35MW 71454563 Ki = 0.057 nM T46185 C6G2HC 71455894 Ki = 1497 nM T46185 CFBC49 71455896 Ki = 5011 nM T46185 CQ98SO 71455965 IC50 = 97.9 nM T46185 CWZ6X0 71455966 IC50 = 58.8 nM T46185 C9N0HT 71455967 IC50 < 5 nM T46185 CS4TY5 71455968 IC50 = 104.7 nM T46185 CLWS62 71455969 IC50 = 548.8 nM T46185 CVI7S2 71457690 Ki = 1488 nM T46185 CP7JI0 71457691 Ki = 552 nM T46185 C3Z9KW 71457770 IC50 = 94.6 nM T46185 C63TRO 71457771 IC50 = 405.1 nM T46185 C56DYG 71457818 IC50 > 3300 nM T46185 CK5T4P 71459604 Ki = 1222 nM T46185 CQ64EL 71459689 IC50 = 178.5 nM T46185 CNKD53 71459690 IC50 < 5 nM T46185 C8Q2FH 71459691 IC50 = 15 nM T46185 CH9R6O 71459724 IC50 = 831.8 nM T46185 C8NWX4 71459909 Ki = 1995.26 nM T46185 COQ67L 71459971 Ki = 17.3 nM T46185 C1CD2B 71461344 Ki > 10000 nM T46185 C2OIW1 71461631 IC50 = 357.1 nM T46185 CG8F1C 71461681 Ki = 3.58 nM T46185 CIP7D8 71462570 Ki = 1.3 nM T46185 CKX5O8 71463061 Ki = 1348 nM T46185 C1Y9IC 71463063 Ki = 1248 nM T46185 CKG3U2 71463133 IC50 > 3300 nM T46185 CCR43M 71463134 IC50 = 998.9 nM T46185 C27RGM 71463135 IC50 = 108.3 nM T46185 C3AKB0 71463136 IC50 = 82.5 nM T46185 C68UAI 71574174 Ki > 100000 nM T46185 C3MJ7B 71575027 Ki = 2030 nM T46185 CN82HY 71575122 Ki > 100000 nM T46185 CY1Q9O 71575447 Ki = 1170 nM T46185 CNS4V8 71575552 Ki > 100000 nM T46185 CM9SQ2 71575553 Ki > 100000 nM T46185 C89MPL 71575652 Ki = 540 nM T46185 CM8UN7 71598549 IC50 > 30000 nM T46185 C1OE9J 71607097 IC50 > 30000 nM T46185 CG75SQ 71741398 Ki = 11.48 nM T46185 C3FQY2 71806339 IC50 > 10000 nM T46185 CEX25Q 72190449 Ki = 1202.26 nM T46185 C79XFZ 72190450 Ki = 407.38 nM T46185 C7NYG0 72190451 Ki = 14454.4 nM T46185 C6PE7F 72190452 Ki = 1548.82 nM T46185 CN4D2K 72191050 Ki < 27542.29 nM T46185 CL1A6K 72191051 Ki < 25703.96 nM T46185 CHE5O6 72545089 Ki > 100000 nM T46185 CI6D4E 72545091 Ki > 100000 nM T46185 CKFW54 72545094 Ki > 100000 nM T46185 CWLO54 72545096 Ki > 100000 nM T46185 C5D4PA 72545098 Ki > 100000 nM T46185 CR39AG 72545326 Ki > 100000 nM T46185 C5HLF7 72545329 Ki > 100000 nM T46185 CWH6T3 72548703 IC50 = 48 nM T46185 CC65OA 73213195 Ki > 10000 nM T46185 CW83DK 73213196 Ki > 10000 nM T46185 C46HUP 73345823 Ki = 116 nM T46185 C4J7PB 73346226 Ki = 7079.46 nM T46185 CUR4F2 73346227 Ki = 912.01 nM T46185 CRG9J8 73346332 Ki = 1732 nM T46185 CK0HR9 73346334 Ki = 1028 nM T46185 CVKN29 73346335 Ki > 10000 nM T46185 C6J0TM 73346336 Ki = 487 nM T46185 C2B1GF 73347725 Ki = 1949.84 nM T46185 CY60RD 73347826 Ki = 2788 nM T46185 CC35AI 73347827 Ki = 2292 nM T46185 C5R1OC 73349360 Ki > 10000 nM T46185 C58SJG 73349591 Ki > 100000 nM T46185 CA6Z1P 73349592 Ki > 100000 nM T46185 C9Z1FO 73350398 Ki = 1340 nM T46185 CBX06Q 73350846 Ki = 19952.62 nM T46185 CDS4F1 73350931 Ki = 474 nM T46185 CA8L9Y 73351145 Ki > 100000 nM T46185 C2TK7H 73352329 Ki = 2238.72 nM T46185 C93IHF 73352330 Ki = 47.86 nM T46185 CV1U7L 73352414 Ki = 1010 nM T46185 C87LGB 73352415 Ki = 1939 nM T46185 CFM9Z0 73353378 Ki = 30.8 nM T46185 C1NJ0R 73353884 Ki = 4414 nM T46185 CL8T4U 73355325 Ki = 2398.83 nM T46185 C4F7VK 73355415 Ki = 195 nM T46185 CA4CP6 73355416 Ki = 8846 nM T46185 C3Z5LT 73355419 Ki = 3553 nM T46185 CX7ZV3 73356454 Ki = 738 nM T46185 CD63YS 73356869 Ki = 151.36 nM T46185 CHV3W1 73774630 EC50 > 30000 nM T46185 C2E7QW 75201901 Ki = 7700 nM T46185 C8IDL3 75306277 Ki > 1000 nM T46185 CC4NP6 75356563 Ki = 6000 nM T46185 C2NE1Q 76309753 IC50 = 687.5 nM T46185 CU5D8H 76309755 IC50 = 1423.4 nM T46185 C42UQX 76309756 IC50 = 1348.8 nM T46185 CO2N6P 76309757 IC50 = 82.5 nM T46185 CZ80LO 76313453 IC50 = 666.4 nM T46185 CFP71X 76313455 IC50 = 1000.3 nM T46185 CNI0G8 76313457 IC50 = 1364.1 nM T46185 CQ2AF0 76316968 IC50 = 638.5 nM T46185 CD3GN5 76316970 IC50 = 253.8 nM T46185 CP7T1M 76320689 IC50 = 519.8 nM T46185 CZ6C0O 76320691 IC50 = 1490.1 nM T46185 CL7U5W 76320693 IC50 = 1404.7 nM T46185 CHZ0P7 76320694 IC50 = 409.8 nM T46185 C94FIP 76324333 IC50 = 228.5 nM T46185 CN2S3T 76324335 IC50 = 2157.2 nM T46185 CA42PY 76324336 IC50 = 190.5 nM T46185 C9ATZ7 76327899 IC50 = 399.8 nM T46185 CQ94CR 76327901 IC50 = 1170.8 nM T46185 CUQ4W3 76327902 IC50 = 467.7 nM T46185 CJFI50 76327903 IC50 = 362.7 nM T46185 CB46FR 76331543 IC50 = 271.2 nM T46185 CXKN87 78319052 EC50 = 2520 nM T46185 C2BM9L 89768534 EC50 > 30000 nM T46185 CB4Y7R 89768546 EC50 > 30000 nM T46185 CYX9R8 89777050 EC50 > 10000 nM T46185 CN0R6C 89777060 EC50 = 2650 nM T46185 C5T3DH 89777147 EC50 > 10000 nM T46185 C5MR9K 89777151 EC50 > 30000 nM T46185 C3MFV0 89777356 EC50 = 1780 nM T46185 C4RUP2 101882890 Ki = 1.698 nM T46185 CC3YS5 118706050 Ki > 100000 nM T46185 C6DXV9 118706052 Ki > 100000 nM T46185 CL4EO9 118706054 Ki = 1737.8 nM T46185 CG86QX 118710659 Ki = 16.22 nM T46185 C9D1MC 118710661 Ki = 5.248 nM T46185 C9H7FI 118710663 Ki = 2.818 nM T46185 CV2JU4 118710665 Ki = 40.74 nM T46185 C97VPM 118710667 Ki = 6.918 nM T46185 CI26PL 118710669 Ki = 3.311 nM T46185 C1OV8Y 118710671 Ki = 2.188 nM T46185 CUV5Y0 118715454 EC50 > 30000 nM T46185 C4JY5S 118719502 IC50 > 30000 nM T46185 CI8CR0 118719920 Ki = 66.07 nM T46185 CV1WX5 118719921 Ki = 10.96 nM T46185 CIAG59 118719922 Ki = 1.38 nM T46185 CC5Q8Y 118719923 Ki = 89.13 nM T46185 CC8R6U 118719924 Ki = 85.11 nM T46185 CT8KO4 118719925 Ki = 3235.94 nM T46185 C16DHZ 118719926 Ki = 602.56 nM T46185 CLA06I 118719927 Ki = 208.93 nM T46185 CF20SR 118719928 Ki = 213.8 nM T46185 C6N7HV 118719929 Ki = 416.87 nM T46185 C64BIA 118719930 Ki = 478.63 nM T46185 CG4ZV5 118719931 Ki = 79.43 nM T46185 C05OBV 118723724 Ki > 100000 nM T46185 C37MUF 118728610 IC50 = 35.1 nM T46185 C96QNO 118728611 IC50 = 6455 nM T46185 CKP85M 122189495 EC50 = 65.4 nM T46185 C2H3QF 122189496 EC50 = 172 nM T46185 C9HG5K 122189499 EC50 = 24 nM T46185 CAJ45R 122190994 EC50 = 749 nM T46185 C7TL4G 122191001 EC50 = 435 nM T46185 CA02ZK 122191002 EC50 = 118 nM T46185 CQI8E1 122191003 EC50 = 211 nM T46185 C80JRU 122191004 EC50 = 411 nM T46185 CF8N0T 122191005 EC50 = 604 nM T46185 C9G0TM 122191006 EC50 = 342 nM T46185 CR93HM 122191007 EC50 = 242 nM T46185 CRF36I 122191008 EC50 = 65.5 nM T46185 C8SDW5 122203596 Ki = 0.7586 nM T46185 CZ61LK 127034966 EC50 > 5011.87 nM T46185 CA0SN5 127034967 EC50 > 5011.87 nM T46185 CJ2O5A 127044078 EC50 > 10000 nM T46185 CJ94GK 129316454 EC50 > 10000 nM T46185 C50GOC 130442480 Ki = 7300 nM T46185 CM04RF 130442572 Ki = 8100 nM T46185 CFXL21 132060812 Ki = 6820 nM T46185 CAVB41 132584404 Ki > 10000 nM T46185 CBU81N 134149168 Ki > 10000 nM T46185 C08GLT 134207682 EC50 = 650 nM T46185 CY24XH 134207690 EC50 = 600 nM T46185 C2X6BZ 134207697 EC50 = 1200 nM T46185 CA16JM 134207728 EC50 > 10000 nM T46185 C1GY2T 135156251 EC50 > 10000 nM T46185 C4UX2M 135430667 Ki = 2187.76 nM T46185 CI5SL0 137633162 EC50 = 27 nM T46185 CVRT14 137633582 Ki = 0.76 nM T46185 CT21NO 137633649 Ki = 0.71 nM T46185 CD91UT 137634680 Ki = 980 nM T46185 COI42G 137635637 EC50 = 239.88 nM T46185 CM9C1Z 137635723 EC50 = 220 nM T46185 C6QB9W 137635734 Ki = 1778.28 nM T46185 CX8O0V 137636308 Ki = 4168.69 nM T46185 CRH92D 137636829 Ki = 15000 nM T46185 CWT0D8 137637047 Ki = 10000 nM T46185 C7VUW4 137637944 IC50 = 330 nM T46185 CY8Q1V 137638270 IC50 = 352 nM T46185 CFDB34 137639384 Ki = 6300 nM T46185 C4YJ1T 137639541 Ki = 46000 nM T46185 CVIA23 137640095 Ki = 5700 nM T46185 CZ4TA9 137640201 Ki = 794.33 nM T46185 CX4A3N 137640511 Ki = 11481.54 nM T46185 C2POD8 137640878 Ki = 27000 nM T46185 C8ZDW1 137642318 Ki = 9200 nM T46185 C4Q6ZM 137642607 Ki = 2398.83 nM T46185 CUDP85 137643254 Ki = 0.41 nM T46185 CW4IJ1 137644950 Ki = 39000 nM T46185 C0KL6Q 137644962 Ki = 4786.3 nM T46185 CPCY48 137645406 Ki = 52 nM T46185 CG8P6I 137645938 Ki = 562.34 nM T46185 CO58KT 137646451 Ki = 630 nM T46185 CN4U1A 137646732 EC50 = 960 nM T46185 CJIU91 137647528 Ki = 29000 nM T46185 C2XMK6 137647734 IC50 = 352 nM T46185 CB9PL0 137648038 Ki = 930 nM T46185 C3LC9W 137648483 Ki = 4400 nM T46185 CBN1K6 137650836 Ki = 0.7079 nM T46185 C6WS1K 137653145 Ki = 14000 nM T46185 CFZS94 137653227 Ki = 50000 nM T46185 CWF8R1 137653324 Ki = 4800 nM T46185 C8XJO5 137653498 Ki = 790 nM T46185 C61WAG 137654353 IC50 = 520 nM T46185 CC7GE8 137654674 EC50 = 10000 nM T46185 CWOV78 137655063 IC50 = 384 nM T46185 CUC54G 137655636 Ki = 204.17 nM T46185 CUKT36 137655796 EC50 = 830 nM T46185 CUZ2V9 137656894 Ki = 1300 nM T46185 CQ2H0S 137657830 Ki = 2400 nM T46185 CWSA41 137658091 Ki = 4200 nM T46185 C6E0JP 137659594 Ki = 140 nM T46185 C4BAP3 137660708 Ki = 22000 nM T46185 C7NJH0 137661079 Ki = 26000 nM T46185 C68QKL 137661317 Ki = 0.1072 nM T46185 CDA8V2 137661377 Ki = 1905.46 nM T46185 C41ZYJ 137701968 EC50 > 30000 nM T46185 C38OTS 145960427 Ki = 199.53 nM T46185 C06LVP 145960466 Ki = 33.11 nM T46185 CSV5D4 145960592 Ki = 95.5 nM T46185 C4KH9G 145960827 Ki = 61.66 nM T46185 CJI6G2 145961125 Ki = 1230.27 nM T46185 CK7OJ5 145961126 Ki = 1548.82 nM T46185 C0XL7S 145961152 Ki = 2290.87 nM T46185 C3WFT9 145961161 Ki = 57.54 nM T46185 CJ50OV 145961495 Ki = 158.49 nM T46185 CAH97Y 145961981 Ki = 426.58 nM T46185 CH1AE6 145962050 Ki = 707.95 nM T46185 CG16NQ 145963288 Ki = 354.81 nM T46185 CWQ46M 145973726 EC50 = 2100 nM T46185 CC2G1V 146025727 Ki = 1700 nM T46185 C6P3SR 153287553 Ki > 10000 nM T46185 CV9G7Z 153287572 Ki > 10000 nM T46185 CO85KL 153287574 Ki > 10000 nM T46185 CY83UA 155511167 Ki = 300 nM T46185 CSR04X 155512177 Ki = 0.69 nM T46185 CCB34Y 155512243 Ki = 7.1 nM T46185 C2BDK6 155513985 Ki = 1.698 nM T46185 C6JSC8 155515662 Ki = 120 nM T46185 CUM2N4 155515982 Ki = 14000 nM T46185 C53FKW 155516382 Ki = 4.266 nM T46185 C0JM8H 155518181 Ki = 220 nM T46185 C0MT4Q 155519740 Ki = 0.2692 nM T46185 CUSA24 155519891 Ki > 10000 nM T46185 C1R9WB 155520414 Ki = 0.72 nM T46185 C3R6GZ 155520947 Ki = 0.49 nM T46185 CPVA65 155521382 Ki = 11.22 nM T46185 CFVP27 155521893 Ki = 0.07943 nM T46185 CL9ET5 155522354 Ki = 1.072 nM T46185 CI2RK6 155523171 Ki = 2.1 nM T46185 CL6O1R 155523647 Ki = 0.1479 nM T46185 C38PTA 155523888 Ki = 7.762 nM T46185 C8V5WM 155524827 EC50 = 250 nM T46185 C5P1YE 155525064 Ki = 22.91 nM T46185 CDQ89Y 155525097 Ki = 0.07943 nM T46185 CBK1S6 155525654 Ki = 0.4 nM T46185 CBK0Y7 155528269 Ki = 12.02 nM T46185 CRPY78 155529196 Ki = 30 nM T46185 CIA9P5 155530272 Ki = 1.4 nM T46185 C1U3VP 155535038 Ki = 9.2 nM T46185 C7CU8J 155535606 Ki = 0.3631 nM T46185 CB79ZW 155536080 Ki > 10000 nM T46185 C2XN8P 155536739 Ki = 100 nM T46185 C9ZW3N 155537081 Ki = 12 nM T46185 CK8G6H 155538050 Ki = 2.692 nM T46185 CW6FY4 155538474 EC50 > 8830 nM T46185 CR17JS 155539026 Ki = 68 nM T46185 C1TKS0 155539410 EC50 = 420 nM T46185 CV2NG9 155539712 Ki = 0.1148 nM T46185 CG3A9Y 155539770 Ki = 1 nM T46185 CMUF93 155540312 Ki = 0.18 nM T46185 CK70MJ 155541812 Ki = 13 nM T46185 C7DMY9 155542295 Ki = 0.11 nM T46185 CL7ZA6 155542839 Ki = 2.6 nM T46185 CS5YB1 155543344 Ki = 9.333 nM T46185 COV93Z 155543943 Ki = 0.3548 nM T46185 CI8KA5 155544834 Ki = 12 nM T46185 C2CB8H 155548585 Ki = 5.37 nM T46185 CMS50Z 155549803 Ki = 2.3 nM T46185 C1UA2M 155550149 Ki = 1.6 nM T46185 C9KBH7 155550435 Ki = 0.07943 nM T46185 CRIJ70 155550631 Ki = 0.0631 nM T46185 CE3F2K 155551015 EC50 > 7350 nM T46185 COF49W 155551902 Ki = 79.43 nM T46185 CX8JA1 155552185 Ki = 17000 nM T46185 C8LRX2 155552304 EC50 > 10000 nM T46185 CXZQ46 155552922 Ki = 46.77 nM T46185 CN4ZH3 155553222 Ki = 0.91 nM T46185 CS1DK6 155554149 Ki = 30 nM T46185 C7TF1D 155554261 Ki = 33.11 nM T46185 C73DFN 155554567 Ki = 0.4266 nM T46185 C1TDY8 155556289 Ki = 0.1738 nM T46185 C2D3SP 155557118 Ki = 19.95 nM T46185 C75PXS 155559290 Ki = 309.03 nM T46185 CEAD84 155559740 Ki = 1.82 nM T46185 CP2U8A 155560012 Ki = 4.169 nM T46185 CU3TF1 155560139 Ki = 1.479 nM T46185 CCO15D 155560304 Ki = 0.2399 nM T46185 CJM85L 155561780 EC50 = 5160 nM T46185 CMX98Q 155562285 Ki = 130 nM T46185 CSO40U 155564307 Ki = 12 nM T46185 CVLR58 155565285 Ki = 239.88 nM T46185 C9AF7I 155565770 Ki = 350 nM T46185 CDS7K2 155566289 Ki = 0.0631 nM T46185 CY30EN 155567379 Ki = 0.07943 nM T46185 C38QRW 155568227 Ki = 21 nM T46185 CKS4A0 155568815 Ki = 1.1 nM T46185 C3N9VU 10251906 Ki > 500 nM T46185 C2O1SZ 168927 EC50 = 436.52 nM T46185 C9RLJ3 3661 Ki = 0.8128 nM T46185 CD6OK3 44455198 Ki = 9 nM T46185 D01UDC 9815331 Ki = 2.6 nM T46185 D02BOW 5926 Ki = 3235.94 nM T46185 D02EXX 3013846 Ki = 630 nM T46185 D02KZD 71598521 IC50 > 30000 nM T46185 D02MJE 10426487 EC50 = 62 nM T46185 D02VGM 23056 Ki = 0.045 nM T46185 D02ZPV 10125445 Ki = 63.1 nM T46185 D03DKZ 42633508 EC50 > 30000 nM T46185 D03RMI 11536903 Ki = 158.49 nM T46185 D04XNH 44318851 Ki = 190 nM T46185 D05EML 21847 IC50 < 1 nM T46185 D05ZUX 44207909 Ki >= 1000 nM T46185 D06IUC 6508730 Ki = 38 nM T46185 D06QRP 5311123 Ki = 1323 nM T46185 D06UXW 107759 Ki = 0.6 nM T46185 D07GPQ 132947 Ki = 0.2692 nM T46185 D09PIN 3378093 Ki > 1000 nM T46185 D09RPR 16737207 Ki > 10000 nM T46185 D0A2KT 3014059 Ki = 23 nM T46185 D0AR0H 6508724 Ki = 55 nM T46185 D0C2DM 9893054 EC50 = 693 nM T46185 D0C9ZE 10105296 Ki = 300 nM T46185 D0F3AN 57664406 Ki = 5495.41 nM T46185 D0F5LH 4634 Ki = 8.1 nM T46185 D0FF6S 16038374 IC50 > 10000 nM T46185 D0G4CG 4629 Ki = 107.15 nM T46185 D0H4BJ 9308 Ki = 25 nM T46185 D0H8XV 12963076 Ki = 1230.27 nM T46185 D0HP1O 119357 Ki = 5.28 nM T46185 D0I9LU 2229 Ki = 87.1 nM T46185 D0IL1B 3494 IC50 = 0.1585 nM T46185 D0JV2S 3008304 EC50 > 30000 nM T46185 D0L1XR 4630 Ki = 17 nM T46185 D0L5MW 181743 Ki > 10000 nM T46185 D0M5ZE 5311416 Ki = 1258.93 nM T46185 D0O9KA 167962 Ki = 31.62 nM T46185 D0P1FJ 71128 Ki = 9.3 nM T46185 D0T2RY 9948320 Ki = 980 nM T46185 D0TX8W 594590 Ki > 19952.62 nM T46185 D0WO3A 4141 Ki = 954.99 nM T46185 D0Z5RQ 656392 IC50 > 5517 nM T46185 D0Z6VT 71737672 EC50 > 30000 nM T65689 D01JUF 5775 Ki = 11.4 nM T65689 D01MDT 5487 Ki = 28.3 nM T65689 D03SKR 2803 Ki = 8.9 nM T65689 D06OFS 68712 Ki = 59.16 nM T65689 D07MOX 439260 Ki > 100000 nM T65689 D09EBS 4636 Ki = 6.194 nM T65689 D0E9PK 4810 IC50 = 3.548 nM T65689 D0K7WK 4595 Ki > 10000 nM T65689 D0L4HY 5702063 Ki = 34.67 nM T65689 D0O6IZ 4436 Ki = 121.6 nM T65689 D0Z2MB 6918107 Ki > 10000 nM T65689 D00OWF 5280953 Ki = 22 nM T65689 C4JQ7T 2068 Ki = 42 nM T65689 COSX53 3519 Ki = 19.01 nM T65689 C32BCH 4656 Ki = 4.797 nM T65689 CL3Q6V 13639 Ki = 39.81 nM T65689 CL34DN 26137 Ki = 1.585 nM T65689 CU86VK 54459 Ki = 7.943 nM T65689 CGW3X5 58533 Ki = 199.53 nM T65689 C3S9TA 58544 Ki = 1.995 nM T65689 C3BQ9D 69591 Ki = 1258.93 nM T65689 CY7ZC9 70319 Ki = 3981.07 nM T65689 CEZ9Q2 71899 Ki = 1.995 nM T65689 C4X7HB 72016 Ki = 52.36 nM T65689 CX17DE 131284 Ki = 231.74 nM T65689 CGT8R0 160510 Ki = 46 nM T65689 CD3ET5 231469 Ki = 7.943 nM T65689 CE5HT0 238079 Ki = 1258.93 nM T65689 COK74Z 345764 Ki = 630.96 nM T65689 C3KM4Y 408156 Ki = 630.96 nM T65689 C4WYR1 594045 Ki = 251.19 nM T65689 C0D5JK 2737433 Ki = 158.49 nM T65689 CUA2H0 3084422 Ki = 31.62 nM T65689 CW04IO 3086495 Ki = 5.012 nM T65689 C1WJ9H 3158580 Ki = 5200 nM T65689 CPCL54 3746427 Ki = 5.012 nM T65689 C98HXL 3771231 Ki = 15.85 nM T65689 C5J1DA 4393018 Ki = 199.53 nM T65689 C6VR5J 6603748 IC50 = 8100 nM T65689 CA51BY 9794143 Ki = 1584.89 nM T65689 C13MBI 9794144 Ki < 10000 nM T65689 C89HIW 9837412 Ki = 10 nM T65689 CB9X7K 9837537 Ki = 1.99 nM T65689 C29SRO 9996353 Ki = 79.43 nM T65689 CUIL41 10012705 Ki = 5.012 nM T65689 C6M4BI 10057802 Ki = 10 nM T65689 CL53TD 10176639 Ki = 537.03 nM T65689 CDOU49 10219780 Ki = 645.65 nM T65689 C0HS9G 10242469 Ki = 7.943 nM T65689 C6Q1DA 10262328 Ki = 10 nM T65689 CL4R3I 10313366 Ki = 512.86 nM T65689 CBYF76 10354045 Ki = 4.7 nM T65689 C5BME0 10374995 Ki = 6.31 nM T65689 C8HWU6 10375456 Ki = 3.162 nM T65689 CUJ32V 10419932 Ki = 11.75 nM T65689 C5DY8H 10442436 Ki = 22.91 nM T65689 CXFE98 10588013 Ki < 10000 nM T65689 C6TFB4 10634173 Ki = 63.1 nM T65689 CF4Y1O 10657832 Ki = 169.82 nM T65689 C0L4QP 10797646 Ki = 331.13 nM T65689 CID3R4 10868559 Ki = 158.49 nM T65689 CZIQ01 10922759 Ki = 10 nM T65689 C8A3LU 10933317 Ki = 470 nM T65689 CT3ZI9 10967219 Ki = 5590 nM T65689 C05XCR 10977777 Ki = 100 nM T65689 CV70ZA 10978438 Ki = 93 nM T65689 CA8Q9Z 10987033 Ki = 1.072 nM T65689 C3VR2W 10997791 Ki = 7244.36 nM T65689 CMU71R 11021868 Ki = 621 nM T65689 CE9T7A 11022127 Ki = 7 nM T65689 C15HYE 11031586 Ki = 3.5 nM T65689 C0A9OC 11031718 Ki = 22.7 nM T65689 CUTM06 11042529 Ki = 31.62 nM T65689 C7Q3ZX 11043404 Ki = 1000 nM T65689 CDIR37 11044324 Ki > 1000 nM T65689 CVB75J 11053968 Ki = 63.1 nM T65689 CJ58RV 11055234 Ki = 560 nM T65689 CJ1QY8 11063180 Ki = 588.84 nM T65689 C0BT2U 11064673 Ki = 43 nM T65689 C5XGY9 11074976 Ki = 10000 nM T65689 CW85AV 11075930 Ki = 140 nM T65689 CT7Q1B 11119320 Ki = 17 nM T65689 CRT6N5 11137887 Ki = 6309.57 nM T65689 CSXV82 11138988 Ki = 47 nM T65689 CGIZ95 11159387 Ki = 6309.57 nM T65689 CL4K0S 11241345 Ki = 50.12 nM T65689 CH2FX9 11747682 Ki = 690 nM T65689 C7LH6B 11770304 Ki = 10000 nM T65689 CAN5Y6 11781522 Ki = 5300 nM T65689 CUB8Q0 12191520 Ki = 100 nM T65689 C78YLK 12248147 Ki = 10000 nM T65689 COYN25 12333190 Ki = 398.11 nM T65689 CPW7N4 12366083 Ki = 10000 nM T65689 C7PEN5 12366096 Ki = 10000 nM T65689 CR1NT6 12632113 Ki = 6025.6 nM T65689 C9GQ4Z 12632114 Ki = 3162.28 nM T65689 CD40XG 12761754 Ki = 3162.28 nM T65689 CKG7B6 12843664 Ki = 7943.28 nM T65689 CNHG28 12863226 Ki = 79.43 nM T65689 CEJ70T 13393069 Ki = 10000 nM T65689 CAK0Y6 13425078 Ki = 50.12 nM T65689 CBTJ50 13425090 Ki = 1584.89 nM T65689 CY97SK 13425094 Ki = 50.12 nM T65689 CMC26O 13869340 Ki = 3.981 nM T65689 C5PD3O 13869343 Ki = 15.85 nM T65689 CQ76WL 14456173 Ki = 10 nM T65689 C7VAQ3 14964720 Ki = 39.81 nM T65689 CCAI21 15407019 Ki = 630.96 nM T65689 CY0NJ5 17774023 Ki = 79.43 nM T65689 C24HWZ 17774025 Ki = 5.012 nM T65689 C8FHS0 17774026 Ki = 39.81 nM T65689 CTD13R 18788392 Ki = 7943.28 nM T65689 CXGA32 19763483 Ki = 158.49 nM T65689 CT84EK 21608213 Ki = 50.12 nM T65689 C2DN1W 21819953 Ki = 25.12 nM T65689 CKIP49 24971933 Ki = 79.43 nM T65689 C21UPD 25883577 Ki = 2.512 nM T65689 C8N7OG 25883581 Ki = 0.7943 nM T65689 CE1Z6D 25883599 Ki = 3.981 nM T65689 C2UX5O 44268929 Ki = 2.512 nM T65689 CZQ54H 44268938 Ki = 1258.93 nM T65689 CO65VL 44269006 Ki = 1.259 nM T65689 C0TP2Z 44269013 Ki = 6.31 nM T65689 CHU5N0 44269016 Ki = 158.49 nM T65689 C5PX3V 44269036 Ki = 63.1 nM T65689 CY01QF 44269044 Ki = 100 nM T65689 C40ZSP 44269051 Ki = 25.12 nM T65689 CUM8P4 44269069 Ki = 10 nM T65689 CR9PJ5 44269074 Ki = 79.43 nM T65689 C6Q8RX 44269086 Ki = 50.12 nM T65689 COB7V3 44269088 Ki = 199.53 nM T65689 CW6A9E 44269089 Ki = 5011.87 nM T65689 C2RWL9 44269090 Ki = 158.49 nM T65689 C7PG8R 44269098 Ki = 398.11 nM T65689 CGQK91 44269099 Ki = 10000 nM T65689 C9T7MG 44269100 Ki = 2.512 nM T65689 CF70OX 44269103 Ki = 79.43 nM T65689 C37XCE 44269105 Ki = 10 nM T65689 CG2D6U 44269106 Ki = 3.981 nM T65689 CPIW69 44269107 Ki = 31.62 nM T65689 CLE3A7 44269115 Ki = 630.96 nM T65689 CZ63DE 44269122 Ki = 309.03 nM T65689 C3I8AT 44269123 Ki = 1995.26 nM T65689 C89FEL 44269124 Ki = 316.23 nM T65689 CFH0C6 44269128 Ki = 3.162 nM T65689 CQZ15X 44269134 Ki = 5011.87 nM T65689 CBS13Z 44269138 Ki = 3162.28 nM T65689 CDS8G5 44269140 Ki = 2511.89 nM T65689 C5SOY3 44269160 Ki = 1000 nM T65689 CN9TV2 44269161 Ki = 39.81 nM T65689 CM57PN 44269162 Ki = 10000 nM T65689 C7V4AB 44302352 Ki > 1000 nM T65689 CS3B6M 44309180 Ki = 17.38 nM T65689 C67ZNM 44352207 Ki = 125.89 nM T65689 CZTA92 44363923 Ki = 37 nM T65689 CIP16C 44403937 Ki = 2022 nM T65689 C13GWS 53821187 Ki = 724.44 nM T65689 CBRI02 78114597 IC50 = 7244.36 nM T65689 CMF3A7 78114671 IC50 = 3388.44 nM T65689 C8JFM6 78114674 IC50 = 8.128 nM T65689 CR6Z8F 78114676 IC50 > 1000000 nM T65689 CTS2P9 78114881 IC50 = 7413.1 nM T65689 C8A6EV 136135852 Ki = 251.19 nM T65689 CAS3E0 155510985 IC50 = 10.47 nM T65689 C75CEX 155513073 IC50 = 1348.96 nM T65689 CVU8Q3 155513359 IC50 = 5495.41 nM T65689 CTV3M6 155521287 Ki = 912000 nM T65689 CK8U7X 155526524 IC50 = 645.65 nM T65689 CD5Y1E 155533747 IC50 = 7585.78 nM T65689 C08RIO 155540329 IC50 = 181.97 nM T65689 CR3T5H 155546767 IC50 = 602559.59 nM T65689 C7V2KX 155547631 IC50 = 28.84 nM T65689 C2EO4B 155567867 IC50 = 64.57 nM T65689 D03LPH 107838 Ki = 180 nM T65689 D04ZPU 11769428 Ki = 0.631 nM T65689 D05GDP 599482 Ki = 12 nM T65689 D05ZUX 44207909 Ki >= 1000 nM T65689 D06BAC 10467319 Ki = 3740 nM T65689 D06QKW 2765 Ki = 3.981 nM T65689 D09BIV 6455104 Ki = 1.995 nM T65689 D09ZDQ 840808 Ki = 2511.89 nM T65689 D0A4AB 2457 Ki = 1.585 nM T65689 D0K8SK 237746 Ki = 5.012 nM T65689 D0LI3J 3080926 Ki = 1.585 nM T65689 D0N9FH 10442227 Ki = 1 nM T65689 D0P4KF 44269078 Ki = 501.19 nM T65689 D0T2RY 9948320 Ki >= 1000 nM T65689 D0Z7NC 33273 Ki = 2.512 nM T82383 D03ZBT 11626560 IC50 < 1 nM T82383 D04KZY 49803313 IC50 < 1 nM T82383 D0IQ6P 25102847 IC50 = 3.4 nM T82383 D0K8KX 5280343 IC50 = 960 nM T82383 D0OB0F 5328940 IC50 = 174 nM T82383 D0R0MW 5329102 IC50 = 9 nM T82383 D00LGR 56839178 EC50 = 222 nM T82383 D03LWG 53235510 IC50 > 10000 nM T82383 D06EGV 44603533 IC50 = 2 nM T82383 D07HPJ 11476171 IC50 > 10000 nM T82383 D0D1GF 42642645 IC50 < 100 nM T82383 D0E3TC 44259 IC50 = 3 nM T82383 D0O6WV 24794418 IC50 = 6 nM T82383 D0T1GF 11282283 IC50 < 1000 nM T82383 D03BNU 59604787 IC50 > 10000 nM T82383 D03RHV 72793043 IC50 = 20800 nM T82383 D08OEW 72792975 IC50 = 1280 nM T82383 D0M9TR 72793042 IC50 = 9890 nM T82383 D0T3ME 156422 IC50 > 30000 nM T82383 C8IAR2 5281657 IC50 > 100000 nM T82383 CI68PW 5283685 IC50 = 32600 nM T82383 CXK0S6 5283727 IC50 = 16900 nM T82383 C4G9WR 9547398 IC50 > 100000 nM T82383 C76CUP 9547698 IC50 = 14700 nM T82383 CR8DA1 10024683 IC50 > 100000 nM T82383 CLA93G 10047202 IC50 = 20200 nM T82383 C3LCH5 10047545 IC50 > 100000 nM T82383 C6M8DY 10285856 IC50 = 10000 nM T82383 C7SFI1 10296883 IC50 = 9100 nM T82383 C4CP7K 10423452 IC50 = 6600 nM T82383 C83QWV 10714343 IC50 = 13100 nM T82383 C8G5WP 11210533 IC50 = 220 nM T82383 C2T8YD 11511361 IC50 = 16 nM T82383 CE5H7D 11544170 IC50 = 182 nM T82383 C69FYK 11604142 Ki = 40 nM T82383 CYL45U 11634544 IC50 = 6 nM T82383 CQ4OC2 11654378 IC50 = 6.4 nM T82383 C64KWZ 11953130 IC50 = 896 nM T82383 C9TU1O 16046126 IC50 > 1000 nM T82383 C9JK2M 16059071 IC50 > 500 nM T82383 CW6UJ9 16059338 IC50 > 300 nM T82383 CH7MS6 16059729 IC50 > 500 nM T82383 CRT0F8 17390026 IC50 > 10000 nM T82383 CR8H4Y 21110084 IC50 > 10000 nM T82383 CA3I4T 24753787 IC50 > 50000 nM T82383 C9B2TF 24880043 IC50 > 1000 nM T82383 CFK2B9 24882503 IC50 > 10000 nM T82383 C5FD1A 24937369 IC50 > 500 nM T82383 C6MP4L 24986245 IC50 = 7 nM T82383 C4AQ3M 24986600 IC50 = 3 nM T82383 CT5NL8 24987305 EC50 = 334 nM T82383 CA4W7M 24987312 IC50 = 2 nM T82383 CS7UK9 24987314 IC50 = 16 nM T82383 CLA59H 24987650 IC50 = 3 nM T82383 C3O9SV 24987652 EC50 = 52 nM T82383 C3DI7Y 24995523 IC50 = 84 nM T82383 CCA6E0 25127414 IC50 = 14 nM T82383 CIUJ83 25167109 IC50 = 389 nM T82383 CIG4H0 25178539 IC50 = 4400 nM T82383 C2TXC6 25218656 IC50 > 500 nM T82383 CVZ09J 42599603 IC50 = 30 nM T82383 CAK0F2 44155856 IC50 < 3 nM T82383 CZKN91 44241537 IC50 = 16 nM T82383 CX4W8V 44252164 IC50 = 77 nM T82383 C53ZWA 44252312 IC50 = 350 nM T82383 CE58PA 44252451 IC50 = 3010 nM T82383 CDHA56 44252599 IC50 = 2600 nM T82383 C8GO1E 44252601 IC50 > 3000 nM T82383 C8HZ7P 44252744 IC50 > 1000 nM T82383 COU84Q 44252746 IC50 > 1000 nM T82383 CEPV43 44252901 IC50 = 6000 nM T82383 CO2K0U 44253336 IC50 = 6400 nM T82383 C1RYE7 44253474 IC50 = 1770 nM T82383 C05BQN 44253476 IC50 = 360 nM T82383 C2S5HZ 44253623 IC50 > 3000 nM T82383 CX7ZP0 44253624 IC50 = 2350 nM T82383 CH2N3Y 44253747 IC50 > 1000 nM T82383 CGY8U9 44253887 IC50 > 1000 nM T82383 C1VT7R 44417767 IC50 = 455 nM T82383 C4ZM1N 44565117 IC50 = 7 nM T82383 CBW2Y1 45268295 IC50 = 524 nM T82383 C0INS5 46194178 IC50 = 10 nM T82383 CF57GK 46215462 IC50 = 14 nM T82383 CYT37A 46232443 IC50 = 14000 nM T82383 C48ZVW 46232555 IC50 = 570 nM T82383 CS9B1U 46232556 IC50 = 430 nM T82383 CDN85C 46870258 IC50 = 58 nM T82383 C30KRS 46870260 IC50 = 100 nM T82383 C8CRK2 49870909 IC50 = 7 nM T82383 CF28WU 50939519 IC50 = 28.9 nM T82383 C38NLV 51049990 IC50 = 18 nM T82383 CE9V5U 52913058 IC50 = 68 nM T82383 CQ2RT1 52913059 IC50 = 1434 nM T82383 CAC9T3 52913870 IC50 = 52 nM T82383 C5HVL9 52914083 IC50 = 72 nM T82383 CH1WR3 52914084 IC50 = 27 nM T82383 CPY2E7 52914189 IC50 = 388 nM T82383 CU3Q4R 52914195 IC50 = 27 nM T82383 CKC41N 52914527 IC50 = 380 nM T82383 C60RVF 52914530 IC50 = 201 nM T82383 C13MUQ 52914647 IC50 = 21 nM T82383 C8W4YA 52914648 IC50 = 121 nM T82383 C30TKO 52914770 IC50 = 430 nM T82383 CM6QE5 52914771 IC50 = 184 nM T82383 C2W9OA 53324451 IC50 > 10000 nM T82383 C3V5XE 53355503 IC50 = 37 nM T82383 C8NA4L 53384644 IC50 > 30000 nM T82383 C8AB1J 54759606 Ki = 63 nM T82383 C9ZFS1 54764923 IC50 = 21900 nM T82383 CC62KV 54915268 IC50 > 10000 nM T82383 CBOD63 56835089 IC50 = 5250 nM T82383 C4S3YK 56839177 IC50 = 19 nM T82383 CPHX64 57325478 IC50 > 50000 nM T82383 CQ9BW4 57325479 IC50 > 50000 nM T82383 CD6Y9Z 57395116 IC50 = 18400 nM T82383 C8W6IG 57395117 IC50 = 23800 nM T82383 CG7S0D 57396882 IC50 = 19400 nM T82383 CJMT39 57597953 IC50 = 4060 nM T82383 CVK0G4 58056356 IC50 > 50000 nM T82383 CC7G1S 58229284 IC50 = 840 nM T82383 C1U6WO 58229285 IC50 = 2250 nM T82383 CDL0P8 58229302 IC50 = 1960 nM T82383 C0O6BL 58229307 IC50 = 1610 nM T82383 C5JG7C 58229331 IC50 = 54 nM T82383 CO9R2K 58229348 IC50 = 31 nM T82383 C41MCI 58229352 IC50 = 300 nM T82383 CK65OM 58229387 IC50 = 35 nM T82383 C3VI7D 58229394 IC50 = 21 nM T82383 CNXU29 58229412 IC50 = 28 nM T82383 C52OMW 58229434 IC50 = 27 nM T82383 C9ZCT2 62705065 IC50 = 446.5 nM T82383 C10AMI 66553589 IC50 > 10000 nM T82383 CM4DT0 66575761 IC50 = 240 nM T82383 C79YEC 66576708 IC50 = 730 nM T82383 C6X8ZG 66576789 IC50 = 440 nM T82383 C2KV4X 66576869 IC50 = 3400 nM T82383 CM26DB 66576870 IC50 = 290 nM T82383 CZS0V9 66576946 IC50 = 420 nM T82383 C3J1FQ 66576947 IC50 = 56 nM T82383 C3XMO7 66576948 IC50 > 10000 nM T82383 C2ZEX1 66929146 EC50 = 47 nM T82383 C9Z6AN 67071363 IC50 = 70 nM T82383 C09VRH 67071376 IC50 = 910 nM T82383 C56QHK 67071384 IC50 = 202 nM T82383 CM34DB 67071387 IC50 = 27 nM T82383 CIK1L9 67071545 IC50 = 101 nM T82383 CD14OC 67071561 IC50 = 51 nM T82383 CTC1N5 67071681 IC50 = 796 nM T82383 CEKN37 67073846 IC50 = 35 nM T82383 CAH4X8 67073886 IC50 = 46 nM T82383 CIN2W1 67073928 IC50 = 636 nM T82383 C72UBJ 67074145 IC50 = 16 nM T82383 CTEN42 67074225 IC50 = 170 nM T82383 C36GAY 67074402 IC50 = 50 nM T82383 CLAZ76 67074403 IC50 = 36 nM T82383 CB5UN2 67074599 IC50 = 21 nM T82383 C6R2LU 67074801 IC50 = 120 nM T82383 CM80BN 67088276 IC50 = 238 nM T82383 CV63UL 67240318 IC50 > 10000 nM T82383 CJLT43 67471113 IC50 = 81 nM T82383 CS35KW 67959157 IC50 = 91 nM T82383 CXR9Y0 68212353 IC50 = 150 nM T82383 CEH69L 68212361 IC50 = 36 nM T82383 C4V3DJ 68212395 IC50 = 50 nM T82383 CPZ8D7 68212421 IC50 = 660 nM T82383 CBUE63 68212479 IC50 = 690 nM T82383 CR0B8N 68212480 IC50 = 12 nM T82383 CZJ83X 68212482 IC50 = 4 nM T82383 C1QXE9 68212489 IC50 = 360 nM T82383 C5H8DO 68212494 IC50 = 17000 nM T82383 C2WDO9 68212498 IC50 = 1400 nM T82383 C7PT2D 68212505 IC50 = 3.7 nM T82383 CKPF54 68212509 IC50 = 1.4 nM T82383 C40GFP 68212528 IC50 = 4600 nM T82383 CJY4P6 68212724 IC50 = 140 nM T82383 C2ZCD6 68212733 IC50 = 38 nM T82383 C4ARE2 68212746 IC50 = 38 nM T82383 CTM2R4 68212750 IC50 = 750 nM T82383 C5MG7K 68212755 IC50 = 180 nM T82383 COV36W 68212757 IC50 = 100 nM T82383 C51DUT 68212759 IC50 = 41 nM T82383 CL95KS 68212760 IC50 = 83 nM T82383 CQD3H2 68212763 IC50 = 610 nM T82383 C6GU4S 68212779 IC50 = 2400 nM T82383 CG5VP7 68212780 IC50 = 380 nM T82383 CJR90K 68212791 IC50 = 59 nM T82383 CS5C0R 68212798 IC50 = 85 nM T82383 C8I7GC 68293638 IC50 > 10000 nM T82383 CD56XK 68293660 IC50 > 10000 nM T82383 CFE1W7 68385049 IC50 = 88 nM T82383 C0CVM4 68853833 IC50 = 15 nM T82383 CDE57I 68854992 IC50 = 3 nM T82383 CRG14Q 68855406 EC50 = 52 nM T82383 CLY7I4 68971880 EC50 = 55 nM T82383 CM4WN5 68976126 EC50 = 52 nM T82383 CWS02A 69268131 EC50 = 62 nM T82383 CH2ME7 69269337 EC50 = 20 nM T82383 CPF8U9 69269522 IC50 = 32 nM T82383 C2S8YO 69270579 IC50 = 4 nM T82383 CMPQ52 69271243 EC50 = 193 nM T82383 C2A7YP 69272308 EC50 = 21 nM T82383 CC5X9W 69272552 IC50 = 10 nM T82383 CB13CE 69272823 EC50 = 16 nM T82383 CQT98L 70681360 IC50 = 2800 nM T82383 CQG1C4 70681387 IC50 = 32 nM T82383 C2B8DE 70681768 IC50 > 30000 nM T82383 CQAU72 70681769 IC50 = 220 nM T82383 CG80HU 70681780 IC50 = 16 nM T82383 CAI38L 70683481 IC50 = 2930 nM T82383 CRE0K6 70683482 IC50 = 61 nM T82383 CTUB80 70683483 IC50 = 37 nM T82383 CLV1A8 70685607 IC50 = 1320 nM T82383 C5F1MS 70685608 IC50 = 3910 nM T82383 CIA8R2 70685609 IC50 = 82 nM T82383 C5F1VZ 70685610 IC50 = 91 nM T82383 CIQ8S5 70685611 IC50 = 1730 nM T82383 C8JYH4 70686029 IC50 = 22000 nM T82383 CER0C7 70687708 IC50 = 6100 nM T82383 C6TGK9 70687737 IC50 = 1630 nM T82383 C4UK0R 70687738 IC50 = 1400 nM T82383 CQR18G 70687739 IC50 = 62700 nM T82383 C62CPH 70689786 IC50 = 1150 nM T82383 CANV90 70689787 IC50 = 1080 nM T82383 C7LVS2 70692345 IC50 = 47 nM T82383 CWP13X 70695379 IC50 > 30000 nM T82383 CM0D3O 70696465 IC50 > 30000 nM T82383 CTB5O3 70696471 IC50 = 57 nM T82383 C5Q3YE 70697396 IC50 > 10000 nM T82383 CH0B8N 70789756 IC50 = 5700 nM T82383 CA3O6K 71552696 IC50 = 61 nM T82383 C1NPL0 71552941 IC50 = 3200 nM T82383 CA4PS8 71552942 IC50 = 3990 nM T82383 C4ITZ0 71717135 IC50 = 27 nM T82383 C4Q2HC 71721525 IC50 = 360 nM T82383 CQ3JN8 71819732 IC50 = 1130 nM T82383 C9NVM8 72192165 IC50 = 260 nM T82383 C7A8XR 72547635 IC50 = 1200 nM T82383 CUPN10 72547636 IC50 = 780 nM T82383 C5MI7D 72547637 IC50 = 610 nM T82383 CD93WQ 72547638 IC50 = 1900 nM T82383 C49RTS 72547864 IC50 > 30000 nM T82383 C45UFT 72547868 IC50 = 7400 nM T82383 CM23ZS 72548104 IC50 = 9000 nM T82383 CO7MN3 72548105 IC50 > 30000 nM T82383 CH05EK 72551069 IC50 = 1700 nM T82383 C07THM 72551070 IC50 = 2000 nM T82383 CVNK29 72551073 IC50 = 400 nM T82383 CO3UW2 72551074 IC50 = 480 nM T82383 CKR0I7 72558179 IC50 = 9 nM T82383 CP09RS 72792559 IC50 > 30000 nM T82383 C3PTC7 72792560 IC50 = 930 nM T82383 C2E0RN 72792562 IC50 = 130 nM T82383 CZXU21 72792563 IC50 = 63 nM T82383 CD7UM4 72792564 IC50 = 72 nM T82383 C38OCL 72792627 IC50 = 61 nM T82383 C39PHS 72792906 IC50 = 170 nM T82383 C6HYA4 72792907 IC50 = 38 nM T82383 C16ETP 72792908 IC50 = 84 nM T82383 CNSX89 72792909 IC50 = 70 nM T82383 C7HXN3 72792910 IC50 > 30000 nM T82383 CGP01I 72792971 IC50 = 550 nM T82383 CXNF57 72792972 IC50 = 180 nM T82383 CGDL83 72792973 IC50 = 830 nM T82383 CJGF34 72792974 IC50 = 1580 nM T82383 C4N9TK 72792977 IC50 = 2790 nM T82383 C5B9CI 72793044 IC50 > 30000 nM T82383 C86UHM 72793045 IC50 > 30000 nM T82383 C75QHA 72793046 IC50 = 3920 nM T82383 C1MPN7 72793047 IC50 = 3530 nM T82383 CRJ81Y 72793048 IC50 = 6180 nM T82383 CL9EA5 72793105 IC50 = 650 nM T82383 CVT7A9 72793106 IC50 = 8040 nM T82383 C39VXU 72793107 IC50 > 30000 nM T82383 C43SNK 72793108 IC50 > 30000 nM T82383 C9XAE8 72793109 IC50 = 20300 nM T82383 CZA34R 72793110 IC50 > 30000 nM T82383 CU9R4X 72793111 IC50 = 430 nM T82383 CD2K0R 72793177 IC50 = 18500 nM T82383 CP26TN 72793178 IC50 = 15000 nM T82383 CKV95R 72793179 IC50 = 3460 nM T82383 CH80BD 72793182 IC50 > 30000 nM T82383 CAJ65L 72793183 IC50 > 30000 nM T82383 CVR1I4 72793252 IC50 = 3000 nM T82383 CJWB46 72793253 IC50 > 30000 nM T82383 CMIH15 72793254 IC50 > 30000 nM T82383 C30IXP 72793255 IC50 = 430 nM T82383 C6YFO5 72793256 IC50 = 560 nM T82383 CJG79M 72793257 IC50 = 580 nM T82383 CK6U5Z 72793332 IC50 = 370 nM T82383 CI6JX5 72793333 IC50 = 16600 nM T82383 CA4ET8 72793334 IC50 = 880 nM T82383 C6JW5N 72793335 IC50 = 1700 nM T82383 CROW51 72793336 IC50 = 3800 nM T82383 C65KJA 72793337 IC50 = 570 nM T82383 C7IA8R 72793397 IC50 = 370 nM T82383 CD85ZE 72793399 IC50 = 530 nM T82383 CI4E7H 72793400 IC50 = 790 nM T82383 C02GET 72793401 IC50 > 30000 nM T82383 C9WYE4 72793466 IC50 = 4700 nM T82383 C37FKG 72793468 IC50 = 10700 nM T82383 COU2I8 72793469 IC50 > 30000 nM T82383 C49MHY 72793532 IC50 = 12600 nM T82383 C3K2BV 72793533 IC50 = 21000 nM T82383 C5UH4O 72793534 IC50 > 30000 nM T82383 C2Z6FI 72793535 IC50 > 30000 nM T82383 CLTB82 72793536 IC50 = 16600 nM T82383 CQ7KX1 72793601 IC50 = 680 nM T82383 CW0PY4 72793602 IC50 = 16200 nM T82383 CKB3O6 72793603 IC50 = 29000 nM T82383 CI9L8K 72793604 IC50 > 30000 nM T82383 CMD9F8 72793605 IC50 = 460 nM T82383 CE60AT 72793606 IC50 = 180 nM T82383 C75UBS 72793607 IC50 = 260 nM T82383 C51VIE 72793608 IC50 = 1100 nM T82383 COL6Y5 72793609 IC50 = 300 nM T82383 CJ9C7M 72793610 IC50 = 5700 nM T82383 CGCL01 72793611 IC50 = 4300 nM T82383 CZ5QY9 72793612 IC50 > 30000 nM T82383 CJ87CG 73211763 IC50 = 270 nM T82383 CVNW01 73386831 IC50 > 1000 nM T82383 C1V3NZ 73425588 IC50 = 1.65 nM T82383 C3UC9H 73891099 IC50 = 160 nM T82383 CQ4ZH2 74538669 IC50 = 120 nM T82383 CG7VE4 76309971 IC50 = 14000 nM T82383 CV8QX0 76310169 IC50 = 6390 nM T82383 CA5L4W 76324771 IC50 = 11000 nM T82383 C17BGH 76328134 IC50 = 3700 nM T82383 C9GO0P 76328313 IC50 = 2460 nM T82383 C39FTZ 76335685 IC50 = 14700 nM T82383 CH8W7D 77461036 IC50 > 1000 nM T82383 CH4OV1 77631108 EC50 = 85 nM T82383 CPG3A5 86302574 IC50 = 8690 nM T82383 CHIZ70 89495685 IC50 = 15 nM T82383 CS6IA4 89495748 IC50 = 32 nM T82383 CW1OS0 89495775 IC50 = 22 nM T82383 CQ2OB9 90292687 IC50 = 448 nM T82383 C29YIS 110474930 IC50 > 10000 nM T82383 C7ZQ0D 110474936 IC50 > 10000 nM T82383 CL2DH6 118433464 IC50 = 218 nM T82383 C01OAD 118433470 IC50 = 213 nM T82383 C9ENZ0 118433703 IC50 = 42 nM T82383 CQU1R4 118443520 IC50 = 560 nM T82383 C8OSQ4 118443521 IC50 = 125 nM T82383 CAM76F 118443524 IC50 = 81 nM T82383 C3DEP2 118443546 IC50 = 118 nM T82383 CGO6B1 118443548 IC50 = 11037 nM T82383 CADG96 118443549 IC50 = 100 nM T82383 CM92EG 118443553 IC50 = 206 nM T82383 CVWR20 118443556 IC50 = 2543 nM T82383 CC9FK0 118443560 IC50 = 64 nM T82383 CRZ68N 118443583 IC50 = 80 nM T82383 C9I5MC 118443585 IC50 = 206 nM T82383 CE42TF 118443586 IC50 = 7356 nM T82383 C5YJT1 118443594 IC50 = 84 nM T82383 CL0YO5 118443595 IC50 = 12.1 nM T82383 CG3K5V 118443597 IC50 = 191 nM T82383 C12WAU 118446433 IC50 = 1690 nM T82383 CFBY13 118446434 IC50 = 26 nM T82383 CQCX41 118737057 IC50 = 578 nM T82383 CY6C1E 122179442 IC50 > 10000 nM T82383 C4X7SD 122192466 IC50 > 10000 nM T82383 COV9E7 124037111 EC50 = 4700 nM T82383 CML3B8 124037112 IC50 = 2.2 nM T82383 C5YT9O 126617627 IC50 = 100 nM T82383 CMA8E0 126617630 IC50 > 10000 nM T82383 CKSX48 126617632 IC50 = 150 nM T82383 C06QEP 126617635 IC50 = 99 nM T82383 CARU63 126617638 IC50 = 560 nM T82383 CA98QM 126617641 IC50 = 78 nM T82383 C6XN4R 126617643 IC50 = 61 nM T82383 CF2Q3D 126617644 IC50 = 30 nM T82383 CD80TV 126617652 IC50 = 230 nM T82383 C8EP1M 126617671 IC50 = 3120 nM T82383 CRYE24 126617672 IC50 > 10000 nM T82383 CBYC49 126617676 IC50 = 4 nM T82383 CUI32Z 126617901 IC50 > 10000 nM T82383 COV36Z 126617902 IC50 = 1890 nM T82383 C8HJ0C 126617903 IC50 = 42 nM T82383 CN1UA8 126617905 IC50 = 26 nM T82383 CIZE72 126617910 IC50 = 200 nM T82383 CFT1Q6 126617917 IC50 = 4377 nM T82383 CDP18S 126617918 IC50 = 888 nM T82383 CQ57KI 126617933 IC50 > 10000 nM T82383 CX2E5B 126617936 IC50 = 530 nM T82383 C85ZHL 126617939 IC50 = 30 nM T82383 C3OX6A 126617945 IC50 > 10000 nM T82383 CH01PO 126617949 IC50 = 620 nM T82383 C6ZK0D 126617966 IC50 = 480 nM T82383 C7GT9H 126617976 IC50 = 78 nM T82383 C2CIT6 126617977 IC50 = 105 nM T82383 CHCM06 126617978 IC50 = 150 nM T82383 CSVH84 126617980 IC50 = 170 nM T82383 C5EU8H 126617983 IC50 > 10000 nM T82383 CINW89 126617985 IC50 > 10000 nM T82383 C1NWO7 126617986 IC50 = 72 nM T82383 C0JBU9 126618285 IC50 = 150 nM T82383 CM6XF4 126618290 IC50 = 6 nM T82383 CS3Y8Q 126618297 IC50 = 74 nM T82383 C5CO7T 126619261 IC50 > 10000 nM T82383 CX60NG 126619264 IC50 > 10000 nM T82383 CDC6W4 126619272 IC50 = 157 nM T82383 C7BM5H 126619273 IC50 = 1120 nM T82383 C1JM0U 126619274 IC50 = 3320 nM T82383 C0A4BG 126619279 IC50 = 34 nM T82383 C8KXV1 127025843 IC50 > 1000 nM T82383 CKS28E 127034802 IC50 = 170 nM T82383 C8ERJ7 127045762 IC50 > 1000 nM T82383 CUO0C5 132156633 IC50 > 10000 nM T82383 CERS64 132937256 IC50 > 30000 nM T82383 C7JC5K 134132904 IC50 = 14 nM T82383 C5DSV1 134134351 IC50 = 390 nM T82383 CYB46P 134135659 IC50 = 620 nM T82383 CDH31O 134136945 IC50 = 11 nM T82383 C46XTD 134138113 IC50 = 340 nM T82383 CK75ZI 134138785 IC50 = 180 nM T82383 CCE1O4 134138988 IC50 = 17 nM T82383 C9V4CG 134140406 IC50 = 120 nM T82383 C5C4TS 134141052 IC50 = 640 nM T82383 CWI41J 134141468 IC50 = 180 nM T82383 CYM06R 134142159 IC50 = 920 nM T82383 CZB68J 134142873 IC50 = 65 nM T82383 CX03CP 134143856 IC50 = 810 nM T82383 C5C2TA 134144975 IC50 = 36 nM T82383 CE12IN 134145489 IC50 = 910 nM T82383 CM4U6L 134147181 IC50 = 26 nM T82383 CBES34 134147807 IC50 = 40 nM T82383 C60FLZ 134148014 IC50 = 18 nM T82383 CDUX09 134148124 IC50 = 1300 nM T82383 CGIT02 134149104 IC50 = 28 nM T82383 C4CA2M 134149641 IC50 = 300 nM T82383 C36GLZ 134150279 IC50 = 4.2 nM T82383 CZ42MI 134150952 IC50 = 110 nM T82383 C39AMZ 134151100 IC50 = 9.3 nM T82383 C10BFN 134151512 IC50 = 170 nM T82383 C8M3RH 134152780 IC50 = 25 nM T82383 C5PV8R 134153049 IC50 = 33 nM T82383 C4M7XF 134153576 IC50 = 120 nM T82383 C4AR9L 134153778 IC50 = 180 nM T82383 C6GC3U 134154700 IC50 = 150 nM T82383 C20PJY 134156194 IC50 = 50 nM T82383 CHN5R6 134156911 IC50 = 93 nM T82383 C70ZRI 134157187 IC50 = 17 nM T82383 C2AN7T 134611886 IC50 > 100000 nM T82383 CYL5V1 134694986 IC50 = 1075 nM T82383 CXC69T 137321158 IC50 = 35 nM T82383 CE75QD 137321162 IC50 = 53 nM T82383 C90YOC 137631907 EC50 = 15 nM T82383 C25ERN 137631967 IC50 > 1000 nM T82383 CORJ86 137632190 EC50 = 39 nM T82383 C3N9PB 137633134 IC50 = 2400 nM T82383 CTZL80 137633249 IC50 = 620 nM T82383 C3TRY8 137634319 IC50 > 10000 nM T82383 CP04EF 137635560 IC50 = 10000 nM T82383 C5T0YN 137636330 IC50 = 9 nM T82383 C06JRX 137637094 IC50 > 1000 nM T82383 CXQ90V 137637834 EC50 = 167 nM T82383 CB6MP3 137638386 EC50 = 216 nM T82383 CB68TY 137638705 IC50 = 1940 nM T82383 C4JOL9 137639535 IC50 = 33 nM T82383 CJ5AV0 137641991 IC50 = 14 nM T82383 C2CGN8 137642165 EC50 = 50 nM T82383 CK67UB 137642879 IC50 = 10200 nM T82383 CZDK13 137643231 IC50 = 89 nM T82383 C1V2MZ 137644127 IC50 > 10000 nM T82383 C8OP1Z 137646065 IC50 = 118 nM T82383 C79HFE 137648309 IC50 > 1000 nM T82383 CR7X6D 137648761 IC50 = 43 nM T82383 CYC6F9 137649379 IC50 > 1000 nM T82383 C35IXH 137650638 IC50 > 1000 nM T82383 C1DK0P 137651391 IC50 > 1000 nM T82383 C8NE0H 137651981 IC50 = 1100 nM T82383 CJ39LQ 137652784 EC50 = 84 nM T82383 CTF2Q9 137653218 IC50 = 3450 nM T82383 CU7R2B 137654115 IC50 > 1000 nM T82383 CO4QM1 137654253 IC50 = 111 nM T82383 CT4XJ1 137654829 IC50 = 2200 nM T82383 CF79VR 137655007 IC50 = 6500 nM T82383 CPKC17 137657071 IC50 = 1800 nM T82383 C45OTU 137657389 IC50 > 630 nM T82383 CVMA26 137657437 IC50 > 1000 nM T82383 CV5H3Z 137657932 IC50 > 1000 nM T82383 C0SJ1X 137658016 IC50 = 210 nM T82383 CSR2O8 137658036 IC50 = 200 nM T82383 CGX4R7 137659569 IC50 > 10000 nM T82383 CO47KH 137659628 IC50 = 130 nM T82383 CLZ08P 137660103 IC50 = 340 nM T82383 CUCS63 137660981 EC50 = 136 nM T82383 CE84NX 144944001 IC50 = 3015 nM T82383 C4HB8M 145949394 IC50 = 62 nM T82383 C65YWX 145964882 IC50 = 260 nM T82383 CHC3T0 145965031 IC50 > 10000 nM T82383 CP92ZF 145965329 IC50 = 120 nM T82383 C9HXI4 145966620 IC50 = 400 nM T82383 CQE9M5 145966810 IC50 = 70 nM T82383 C1EH6C 145967078 IC50 = 1300 nM T82383 CWJ12M 145969155 IC50 = 13 nM T82383 CGW5S1 145969844 IC50 = 380 nM T82383 CB8R3A 145970271 IC50 = 7200 nM T82383 C40VIL 145972979 IC50 = 530 nM T82383 CQBY19 145974023 IC50 > 10000 nM T82383 C4X7CT 145977420 IC50 = 760 nM T82383 CLA57T 145978300 IC50 = 780 nM T82383 C6KDQ5 145979093 IC50 = 3295 nM T82383 CV7QY8 145981517 IC50 = 230 nM T82383 CG0R3A 145984368 IC50 = 0.77 nM T82383 CV78XO 145985621 IC50 = 3291 nM T82383 C03PYD 145986466 IC50 < 1000 nM T82383 CX5MB2 145986730 IC50 = 1084 nM T82383 C1V6RA 145988134 IC50 > 100000 nM T82383 CD98JK 145989189 IC50 = 340 nM T82383 CWH69B 145989428 IC50 = 161 nM T82383 CZCS58 145989494 IC50 = 79 nM T82383 C0PHA7 145990595 IC50 = 70 nM T82383 CN6T4K 145991513 IC50 = 2000 nM T82383 CMBH76 145991936 IC50 = 15 nM T82383 C0SO4N 145993259 IC50 = 416 nM T82383 CI7F4G 145994227 IC50 = 152 nM T82383 C5JN1C 146834963 IC50 = 1.6 nM T82383 CL4UK2 147025626 IC50 = 2.5 nM T82383 C0QS4R 147462141 IC50 = 4.5 nM T82383 CMTD91 149448370 IC50 = 1.2 nM T82383 CF25LS 152815814 IC50 = 10.3 nM T82383 C7EXW9 155510641 IC50 > 20000 nM T82383 CJ1WY3 155510993 IC50 > 20000 nM T82383 C2MD1Q 155513187 IC50 > 10000 nM T82383 C28YIV 155515296 IC50 = 890 nM T82383 CP0U7G 155516158 IC50 = 354 nM T82383 CX1Y3R 155517692 IC50 > 20000 nM T82383 CAR90E 155518004 IC50 = 4.5 nM T82383 CCWR27 155518146 IC50 = 0.94 nM T82383 C52VES 155519524 IC50 = 9100 nM T82383 CQW21U 155520733 IC50 > 1000 nM T82383 CR40TA 155525863 IC50 = 80 nM T82383 CMU83P 155528015 IC50 = 2900 nM T82383 CMAL65 155528486 IC50 > 20000 nM T82383 C71VBU 155528815 IC50 = 93 nM T82383 C67UCP 155529095 IC50 = 126 nM T82383 C8YBM7 155530002 IC50 > 20000 nM T82383 CZ6HQ1 155530683 IC50 = 192 nM T82383 CN8JX1 155536147 IC50 = 2600 nM T82383 CZF86O 155537833 IC50 > 20000 nM T82383 C9MO0L 155537855 IC50 = 216 nM T82383 CTSM92 155538441 IC50 < 0.5 nM T82383 C0ALP9 155540176 IC50 = 0.7 nM T82383 C7H2MN 155542059 IC50 > 20000 nM T82383 CN5EX8 155542818 IC50 = 289 nM T82383 C9PMC5 155546111 IC50 > 20000 nM T82383 CEWS62 155552568 IC50 > 20000 nM T82383 C8EJ7L 155552991 IC50 > 20000 nM T82383 C48BCV 155553696 IC50 = 790 nM T82383 C3TQR9 155554845 IC50 > 30000 nM T82383 CVM2Q4 155555829 IC50 > 20000 nM T82383 CFY52U 155555877 IC50 > 20000 nM T82383 C26MZK 155557683 IC50 = 1500 nM T82383 C43LYT 155561169 IC50 = 8.3 nM T82383 C40IYS 155562258 IC50 = 8.2 nM T82383 C0Y7NL 155568698 IC50 = 218 nM T82383 C1DJN0 155569415 IC50 = 356 nM T82383 D06HVH 54613583 IC50 > 10000 nM T82383 D09TFN 56847486 IC50 = 19 nM T82383 D0L3JR 25212148 IC50 = 1.5 nM T82383 D0N4LR 53469448 IC50 = 2705 nM T82383 D0Y4BL 11676971 IC50 = 12 nM T00156 D04AIT 5280445 IC50 > 10000 nM T00156 D0K8KX 5280343 IC50 = 6500 nM T00156 C3XJB2 17466271 IC50 = 4000 nM T00156 C81ITX 85473309 IC50 = 0.52 nM T00156 C4O1LQ 85473438 IC50 = 1.3 nM T00156 CN0LY2 118863086 IC50 <= 21 nM T00156 C2K8QX 118863093 IC50 <= 21 nM T00156 CB4NJ6 118863095 IC50 <= 21 nM T00156 C3ZID9 118863096 IC50 <= 21 nM T00156 C9KG7L 118863100 IC50 <= 21 nM T00156 C2F3TH 118863101 IC50 <= 21 nM T00156 C30MGC 118863111 IC50 <= 21 nM T00156 CI1V0B 118863115 IC50 <= 21 nM T00156 C2Q0DM 118863117 IC50 <= 21 nM T00156 CE3R7L 118863118 IC50 <= 21 nM T00156 CC2MX3 118863119 IC50 <= 21 nM T00156 C69VME 118863121 IC50 <= 21 nM T00156 C49YNF 118863125 IC50 <= 21 nM T00156 CD47VT 118863126 IC50 <= 21 nM T00156 C2IR3X 118863130 IC50 <= 21 nM T00156 CJZW34 118863134 IC50 <= 21 nM T00156 C8H1JU 118863138 IC50 <= 21 nM T00156 C5R0GU 118863139 IC50 <= 21 nM T00156 CH08RQ 118863140 IC50 <= 21 nM T00156 C1LC3X 118863144 IC50 <= 21 nM T00156 CG28TF 118863146 IC50 <= 21 nM T00156 C3O1NY 118863150 IC50 <= 21 nM T00156 CPN6B0 118863151 IC50 <= 21 nM T00156 C70FVE 118863767 IC50 = 408 nM T00156 CEK8W9 118863773 IC50 = 408 nM T00156 CSL35F 118863775 IC50 = 408 nM T00156 C21UMR 118863776 IC50 = 408 nM T00156 CYUA53 118863780 IC50 = 408 nM T00156 CI0Q8O 118863789 IC50 = 408 nM T00156 CAV6D2 118869687 IC50 < 1 nM T00156 CWY07H 118869698 IC50 <= 1 nM T00156 C0A5LF 118869701 IC50 <= 1 nM T00156 C8EIH9 118869702 IC50 <= 1 nM T00156 CSD4J9 118869706 IC50 <= 1 nM T00156 CM6BU3 118869709 IC50 < 1 nM T00156 CXHM06 118869716 IC50 <= 1 nM T00156 C6PZE4 118871740 IC50 = 408 nM T00156 C3R5FM 118871742 IC50 = 408 nM T00156 CA83VR 118873088 IC50 <= 1 nM T00156 CIS83W 118874989 IC50 = 195 nM T00156 C1WV4E 118874990 IC50 = 195 nM T00156 C72SKO 118874991 IC50 = 195 nM T00156 CMR3T2 118874993 IC50 = 195 nM T00156 CGXH82 118875024 IC50 = 195 nM T00156 CIU8D0 118875025 IC50 = 195 nM T00156 CW39SE 118875317 IC50 = 195 nM T00156 C5OJ9A 118875472 IC50 >= 14 nM T00156 CS98NA 118875482 IC50 >= 14 nM T00156 C17QPT 118875484 IC50 >= 14 nM T00156 C1LM0R 118875489 IC50 >= 14 nM T00156 C0BO4T 118875492 IC50 >= 14 nM T00156 CDK24J 118875495 IC50 >= 14 nM T00156 CPXH61 118875498 IC50 >= 14 nM T00156 CO7DH4 118875501 IC50 >= 14 nM T00156 CRDN23 118875502 IC50 >= 14 nM T00156 CZY36Q 118875503 IC50 >= 14 nM T00156 CPR1D2 118875505 IC50 >= 14 nM T00156 CNE3I8 118875507 IC50 >= 14 nM T00156 CMYF76 118875508 IC50 >= 14 nM T00156 C1J7NZ 118875513 IC50 >= 14 nM T00156 CSGY54 118875515 IC50 >= 14 nM T00156 CD06VZ 118875519 IC50 >= 14 nM T00156 CPR06U 118875521 IC50 >= 14 nM T00156 COT70M 118875523 IC50 >= 14 nM T00156 C0ZU9Q 118875529 IC50 >= 14 nM T00156 C3DR2H 118875530 IC50 >= 14 nM T00156 CHG50S 118875531 IC50 >= 14 nM T00156 CWD0N5 118875534 IC50 >= 14 nM T00156 C2OJ5K 118875536 IC50 >= 14 nM T00156 C5BP2E 118875537 IC50 >= 14 nM T00156 C1A0QV 118875539 IC50 >= 14 nM T00156 CL8AG4 118875542 IC50 >= 14 nM T00156 C2BU4Z 118875546 IC50 >= 14 nM T00156 C1C5JI 118875551 IC50 >= 14 nM T00156 CT45LE 118875552 IC50 >= 14 nM T00156 CFT6A7 118875556 IC50 >= 14 nM T00156 CRFO25 118875896 IC50 >= 14 nM T00156 C2P4ZO 118881830 IC50 = 23.3 nM T00156 C7RO0H 118886841 IC50 = 195 nM T00156 C8C7TF 133638366 IC50 = 18000 nM T00156 CL0EM9 137553166 IC50 = 280 nM T00156 C53WBO 138471562 IC50 = 1900 nM T00156 CG3NZ9 138471719 IC50 > 30000 nM T00156 C81ILP 138471783 IC50 = 180 nM T00156 CR8Y6X 138471822 IC50 = 27000 nM T00156 CK74TQ 138471823 IC50 = 1900 nM T00156 CY0X5W 138471830 IC50 > 30000 nM T00156 CNA9B0 138472065 IC50 = 2400 nM T00156 CTY2K7 138472070 IC50 > 30000 nM T00156 CASK71 138472116 IC50 = 500 nM T00156 CU21NW 138472270 IC50 = 28000 nM T00156 C7AST5 138472335 IC50 = 1800 nM T00156 C8PEM2 138472351 IC50 = 490 nM T00156 C0IT5K 138483587 IC50 = 380 nM T00156 C4D2PC 138483600 IC50 = 8000 nM T00156 CHQ08P 138483659 IC50 = 1500 nM T00156 CZ5XI7 138483744 IC50 = 650 nM T00156 CQMK18 138483746 IC50 = 530 nM T00156 CY3RQ2 138483771 IC50 = 9600 nM T00156 CL3P0U 138483778 IC50 > 30000 nM T00156 C91XCD 138483781 IC50 = 660 nM T00156 C2IE3R 138483782 IC50 > 30000 nM T00156 CZ1MA7 138483783 IC50 > 30000 nM T00156 CS2FM8 138483817 IC50 > 30000 nM T00156 CEKR42 138483818 IC50 = 650 nM T00156 CZ75AN 138483832 IC50 = 14500 nM T00156 CJ82UC 138483850 IC50 = 530 nM T00156 C2R3SV 138484037 IC50 = 11200 nM T00156 C1QIU9 138484162 IC50 > 30000 nM T00156 CDO1P4 138484378 IC50 > 30000 nM T00156 CEK6B1 139300630 IC50 > 10000 nM T00156 C97AHK 142546650 IC50 = 8800 nM T00156 C4S9EI 155519644 IC50 > 30000 nM T00156 C2RX4W 155527140 IC50 = 8200 nM T00156 C4D3EO 155535251 IC50 = 2800 nM T00156 C7YU6M 155536492 IC50 = 11000 nM T00156 CUR4E5 155538216 IC50 <= 1 nM T00156 CFM75S 155544430 IC50 = 27000 nM T00156 CR2P9O 155551823 IC50 = 16000 nM T00156 CX3BT1 155557388 IC50 > 30000 nM T00156 CRSD12 155560733 IC50 > 30000 nM T00156 D00RIX 5280443 IC50 > 10000 nM T00156 D0G3TK 5280863 IC50 = 3900 nM T00156 D0JV2P 2455 IC50 = 300 nM T00156 D0T3PW 5281672 IC50 > 10000 nM T00156 D0Y7HG 5281616 IC50 = 450 nM T69619 D0P9AC 3675 IC50 = 19.95 nM T69619 D03TFJ 5798 IC50 > 100000 nM T69619 D01LAC 6437850 IC50 = 20 nM T69619 C5PSY3 6183 IC50 = 58.88 nM T69619 C3BCZ5 8706 IC50 > 100000 nM T69619 CTJ0C5 13624 IC50 = 4100 nM T69619 C0YU1V 16157 IC50 > 100000 nM T69619 C16YST 21954 IC50 = 20 nM T69619 C6X7TQ 45450 IC50 = 64.57 nM T69619 CQ7E9B 74187 IC50 > 100000 nM T69619 C78YPS 80495 IC50 > 100000 nM T69619 CNK5J2 122074 IC50 = 74000 nM T69619 C1HY2B 135136 IC50 > 100000 nM T69619 CD89VU 137235 IC50 > 100000 nM T69619 CDK18F 198458 IC50 = 269.15 nM T69619 CN6YG0 519332 IC50 > 100000 nM T69619 CQD2N8 728567 IC50 > 100000 nM T69619 CX30AP 2723957 IC50 > 100000 nM T69619 CVSU04 9817917 IC50 = 230 nM T69619 CP0U6F 9834313 IC50 = 407.38 nM T69619 CPE4X0 9836390 IC50 = 309.03 nM T69619 CMC37G 9838666 IC50 = 208.93 nM T69619 CCNY29 9899578 IC50 = 330 nM T69619 C9C6LU 10334080 IC50 = 150 nM T69619 C7X8OB 10344711 IC50 = 20 nM T69619 CCUJ60 10445232 IC50 = 5000 nM T69619 CY41LT 10445774 IC50 = 170 nM T69619 C9X2AQ 10583188 IC50 = 1700 nM T69619 CBP6U9 10589155 IC50 = 1600 nM T69619 COG41X 10619341 IC50 = 2100 nM T69619 CDY0H7 10728071 IC50 = 130 nM T69619 C9ILF3 11147919 IC50 = 100000 nM T69619 CUL1G2 11171749 IC50 = 56000 nM T69619 CI2ZB6 11182637 IC50 = 8000 nM T69619 CV0MO3 11184629 IC50 = 16000 nM T69619 C7QW3P 11229730 IC50 = 79000 nM T69619 C25MKL 11263687 IC50 > 100000 nM T69619 C9OU4R 11321047 IC50 = 2000 nM T69619 CQV28Z 11333471 IC50 = 5600 nM T69619 C3AYC4 11366979 IC50 = 16000 nM T69619 C2BV6C 11508380 IC50 = 19 nM T69619 CKV38A 11655814 IC50 = 53 nM T69619 COU09A 12655267 IC50 > 100000 nM T69619 CI9G2Y 12733693 IC50 > 100000 nM T69619 CDG8V5 12776702 IC50 = 346.74 nM T69619 C3H0EY 14933021 IC50 > 100000 nM T69619 CT8H1K 16206718 IC50 = 181.97 nM T69619 CZGJ10 17778061 IC50 = 323.59 nM T69619 CM8TD3 19926386 IC50 = 109.65 nM T69619 CH56AF 20668674 IC50 > 100000 nM T69619 CUV62I 21361090 IC50 = 416.87 nM T69619 CY79MI 21361101 IC50 = 346.74 nM T69619 CD47FT 21361102 IC50 = 269.15 nM T69619 CAB57Y 21361103 IC50 = 281.84 nM T69619 C9GAP5 21361104 IC50 = 309.03 nM T69619 CY6LZ9 21361108 IC50 = 562.34 nM T69619 C8U7CH 21361111 IC50 = 52.48 nM T69619 CHM46D 21361112 IC50 = 28.84 nM T69619 CUE4T0 21361113 IC50 = 1200 nM T69619 CZV8H4 21914708 IC50 = 1100 nM T69619 C4BCT0 21914733 IC50 = 210 nM T69619 CMX15U 21914735 IC50 = 520 nM T69619 C40JVY 21914801 IC50 = 11000 nM T69619 CMU31P 21914814 IC50 > 100000 nM T69619 C1F7WE 21914821 IC50 = 36 nM T69619 C7WSI5 21914878 IC50 = 730 nM T69619 C8XJ6F 21914885 IC50 = 5000 nM T69619 CKRJ38 21914897 IC50 = 160 nM T69619 CZ1LD4 21914902 IC50 = 9600 nM T69619 CJ4FR2 21914923 IC50 = 3000 nM T69619 CQTS58 21914947 IC50 = 330 nM T69619 C35DAL 21915003 IC50 = 34 nM T69619 CIX98T 21915149 IC50 = 1100 nM T69619 CMI14L 21915171 IC50 = 680 nM T69619 CFT7K9 21915271 IC50 > 10000 nM T69619 CB0K6U 21915298 IC50 = 3500 nM T69619 CLY3Z2 21915304 IC50 = 320 nM T69619 CTO31X 23033764 IC50 = 239.88 nM T69619 CK8R7C 24952865 IC50 > 100000 nM T69619 CK8A4U 25029056 IC50 = 32000 nM T69619 CFYI84 42601491 IC50 = 20 nM T69619 C7HG2X 42623114 IC50 = 260 nM T69619 CUEJ23 42623116 IC50 = 370 nM T69619 CT9LN0 42623192 IC50 = 140 nM T69619 C8EK3R 42623200 IC50 = 30 nM T69619 CJ4MD2 42623269 IC50 = 10 nM T69619 CCAW14 42623272 IC50 = 40 nM T69619 CQ40TO 42623611 IC50 = 180 nM T69619 C5N7SE 42624010 IC50 = 290 nM T69619 CT1ND7 42624011 IC50 = 40 nM T69619 CN96DS 42624091 IC50 = 160 nM T69619 CXU9W0 42624092 IC50 = 1070 nM T69619 C6WVE8 42624093 IC50 = 190 nM T69619 C1QAC5 42624094 IC50 = 70 nM T69619 C7SE6I 42624095 IC50 = 210 nM T69619 CZ0T8M 42624097 IC50 = 150 nM T69619 CPB14W 42624186 IC50 = 80 nM T69619 CKY5J6 42624187 IC50 = 20000 nM T69619 CEF0Y7 42624190 IC50 = 240 nM T69619 CCGY96 42624286 IC50 = 20 nM T69619 CMBT65 44387943 IC50 = 100000 nM T69619 CO6A3U 44387955 IC50 = 3200 nM T69619 C3ZRO0 44387981 IC50 = 440 nM T69619 C2YI1D 44387984 IC50 = 20 nM T69619 CZJY25 44387994 IC50 > 100 nM T69619 C2H1UN 44387996 IC50 = 350000 nM T69619 CH0W8E 46929424 IC50 = 257.04 nM T69619 CI67ZW 46929632 IC50 = 323.59 nM T69619 CZE25T 46929633 IC50 = 218.78 nM T69619 CZ7MD1 46929634 IC50 = 199.53 nM T69619 CC8A0K 46929635 IC50 = 426.58 nM T69619 C1NG9K 46929733 IC50 = 257.04 nM T69619 CUE87S 46929734 IC50 = 257.04 nM T69619 C2P6CA 46929845 IC50 = 436.52 nM T69619 C1RE7I 46929846 IC50 = 575.44 nM T69619 CN81AZ 46929847 IC50 = 407.38 nM T69619 C40NJT 46929848 IC50 = 426.58 nM T69619 CZ02YI 46929849 IC50 = 323.59 nM T69619 CM6P1Z 46929944 IC50 = 630.96 nM T69619 C49WSZ 46929945 IC50 = 398.11 nM T69619 CLN92K 46929946 IC50 = 229.09 nM T69619 C1ZE5B 46929948 IC50 = 346.74 nM T69619 CTR17A 46929950 IC50 = 389.05 nM T69619 CL2JQ1 46929953 IC50 = 91.2 nM T69619 C4T8PH 46929955 IC50 = 109.65 nM T69619 C3AL5C 46929957 IC50 = 169.82 nM T69619 C5V8CB 46930049 IC50 = 120.23 nM T69619 CF5M8A 46930051 IC50 = 70.79 nM T69619 CI7O6F 46930053 IC50 = 346.74 nM T69619 CD10EM 46930055 IC50 = 89.13 nM T69619 CT1O6E 46930057 IC50 = 60.26 nM T69619 C37WIY 46930059 IC50 = 371.54 nM T69619 CMZ5C7 46930061 IC50 = 346.74 nM T69619 CQAO23 46930063 IC50 = 331.13 nM T69619 CB4VE9 46930148 IC50 = 79.43 nM T69619 CHGT58 46930150 IC50 = 2238.72 nM T69619 CQV39D 46930152 IC50 = 436.52 nM T69619 C9I2QR 52937516 IC50 = 50000 nM T69619 CUYB57 52937518 IC50 = 40 nM T69619 CJGN43 52937519 IC50 = 150 nM T69619 CK2L6I 52937625 IC50 = 280 nM T69619 CQ0L9P 52937626 IC50 = 1180 nM T69619 CI73HU 52937627 IC50 = 1060 nM T69619 CEFT21 52945459 IC50 = 467.74 nM T69619 CRI63H 59004572 IC50 = 150 nM T69619 CT8L4F 59004578 IC50 = 8800 nM T69619 C1HS5X 59588962 IC50 = 250 nM T69619 C3NFG6 59588969 IC50 = 40 nM T69619 CY54PA 60172362 IC50 = 71 nM T69619 C9GZD0 60198957 IC50 = 290 nM T69619 C52JYI 65439716 IC50 = 82000 nM T69619 CL7WS5 68106325 IC50 = 31 nM T69619 CCM7E3 68106541 IC50 = 340 nM T69619 C6N9XV 68106705 IC50 = 240 nM T69619 CS50OY 68107525 IC50 = 25 nM T69619 CG08PY 70683622 IC50 > 100000 nM T69619 CHY0R1 71525098 IC50 = 22000 nM T69619 CNH81D 71525102 IC50 = 42000 nM T69619 C7AB4S 71525141 IC50 = 1100 nM T69619 CJ0DP2 71525142 IC50 > 100000 nM T69619 C8VN5H 71525144 IC50 = 18000 nM T69619 CR95DH 71525188 IC50 = 15000 nM T69619 CR56JF 71602638 IC50 = 390 nM T69619 CZH46Y 71713909 IC50 = 13000 nM T69619 C1IA9P 71713912 IC50 = 2200 nM T69619 CAV92G 71812246 IC50 = 5 nM T69619 CG0JN8 72793902 IC50 = 20 nM T69619 CG10MU 89600638 IC50 = 47 nM T69619 CR4DI8 89600723 IC50 = 9.2 nM T69619 C5U0ZG 117949685 IC50 = 50.12 nM T69619 CCG05U 117949686 IC50 > 3162.28 nM T69619 C84UJE 130302628 IC50 > 30000 nM T69619 C3M2IV 130344977 IC50 = 1300 nM T69619 CE8Q7I 130345035 IC50 = 48000 nM T69619 C01UGK 130345060 IC50 = 3600 nM T69619 CN9S7B 130345097 IC50 = 47100 nM T69619 C3CH7B 130345110 IC50 = 19600 nM T69619 C7RN8L 130345158 IC50 >= 100000 nM T69619 CF20BS 130345178 IC50 = 1200 nM T69619 CMO50A 130345200 IC50 = 49000 nM T69619 C29WVS 130358344 IC50 = 74300 nM T69619 CZM13E 130358354 IC50 = 36300 nM T69619 CA8OT9 134135554 IC50 = 4100 nM T69619 C7TPW0 134137520 IC50 = 3000 nM T69619 CDS0V2 134137932 IC50 > 100000 nM T69619 CT17KV 134138256 IC50 = 1600 nM T69619 CB9C2H 134138777 IC50 = 480 nM T69619 C1HY7Z 134140283 IC50 = 560 nM T69619 CVOF10 134140491 IC50 = 180 nM T69619 CVY8I5 134141357 IC50 = 1800 nM T69619 CH1CF7 134142045 IC50 > 100000 nM T69619 C9R0MJ 134142669 IC50 = 2000 nM T69619 C4Q1IF 134143172 IC50 = 610 nM T69619 C0DGI5 134143197 IC50 = 460 nM T69619 CS18EX 134144415 IC50 = 4000 nM T69619 C4RD6O 134145917 IC50 > 100000 nM T69619 CUV96D 134146082 IC50 = 280 nM T69619 CYJ9S8 134146322 IC50 > 100000 nM T69619 CSGB51 134147377 IC50 = 800 nM T69619 C6WZ0N 134147690 IC50 = 420 nM T69619 CJ32HY 134149882 IC50 = 83 nM T69619 C2GRV7 134151663 IC50 = 14000 nM T69619 C5TVY0 134153560 IC50 = 1300 nM T69619 CU5R4T 134155775 IC50 = 330 nM T69619 C0KJZ5 134157682 IC50 > 100000 nM T69619 C9P4YE 137459864 IC50 = 7943.28 nM T69619 CL7HO6 137631916 IC50 > 10000 nM T69619 CR1VX3 137634929 IC50 = 300 nM T69619 CFE6J7 137638698 IC50 = 240 nM T69619 CHYF05 137642678 IC50 = 2000 nM T69619 CH5TK8 137644399 IC50 = 5100 nM T69619 CX1ZT6 137646481 IC50 = 45 nM T69619 C2GF5W 137648175 IC50 > 10000 nM T69619 C4JC8F 137649505 IC50 = 250 nM T69619 C1Z2MU 137649566 IC50 = 31 nM T69619 CJ2N6G 137651583 IC50 = 24 nM T69619 C3RMF4 137653859 IC50 = 55 nM T69619 CG8WJ0 137656048 IC50 = 130 nM T69619 CPG6W2 137657508 IC50 = 1500 nM T69619 CE6P2M 137660742 IC50 = 1700 nM T69619 C6NG3C 137660775 IC50 = 140 nM T69619 CN5JD9 146029690 IC50 = 600 nM T69619 C8QOT7 146029691 IC50 = 31 nM T69619 CT3YI7 146029692 IC50 = 24 nM T69619 CGS13B 146029978 IC50 = 25 nM T69619 C0PL4R 146029979 IC50 = 56 nM T69619 CZ25CL 146029980 IC50 = 54 nM T69619 CZRX72 146029981 IC50 = 410 nM T69619 CHX97R 146029982 IC50 = 400 nM T69619 C35QIR 146029983 IC50 = 160 nM T69619 C5E4LF 146029984 IC50 = 110 nM T69619 C0K5TI 146029985 IC50 = 140 nM T69619 CO04TY 146029986 IC50 = 45 nM T69619 CI6W8F 146029987 IC50 = 40 nM T69619 CFV8M1 146029988 IC50 = 530 nM T69619 C4VNE5 146029989 IC50 = 99 nM T69619 CS7K9F 146029990 IC50 = 77 nM T69619 C7H4LQ 146029991 IC50 = 13 nM T69619 C2V0WM 146029992 IC50 = 17 nM T69619 CI0V5F 155525579 IC50 = 13300 nM T69619 CCN0P3 155545992 IC50 > 31622.78 nM T69619 CWL16Z 155550534 IC50 > 100000 nM T69619 CA35OS 155560404 IC50 > 31622.78 nM T69619 COF96P 155564105 IC50 > 100000 nM T00820 D0X7HV 177852 EC50 = 436.52 nM T00820 CEUK24 581330 EC50 = 276 nM T00820 CK1SB8 4397986 EC50 = 18 nM T00820 CC1R3V 9982698 EC50 = 194 nM T00820 CZQ4S2 10005749 EC50 > 10000 nM T00820 CQ5IA6 10021851 EC50 = 137 nM T00820 CBL2G4 10022595 EC50 = 131 nM T00820 CB9ER0 10045948 EC50 = 45 nM T00820 CWM9N1 10048301 EC50 = 5310 nM T00820 CHQO01 10068147 EC50 = 72 nM T00820 C5CGX3 10071165 EC50 = 5550 nM T00820 C12SXU 10073922 EC50 = 84 nM T00820 C4F1MI 10074379 EC50 = 80 nM T00820 CNQ9V1 10090361 EC50 = 2220 nM T00820 CN47CU 10092671 EC50 = 495 nM T00820 CJ8SB4 10092786 EC50 = 4340 nM T00820 CYA8K7 10114127 EC50 = 1698.24 nM T00820 CST2B3 10115466 EC50 = 6025.6 nM T00820 CN8M5O 10117487 EC50 = 812.83 nM T00820 C75NAR 10118048 EC50 = 537.03 nM T00820 C3WGL0 10159877 EC50 = 2754.23 nM T00820 CYOP70 10160667 EC50 = 1288.25 nM T00820 CR8WV4 10163703 EC50 = 1174.9 nM T00820 CSGK21 10183008 EC50 = 457.09 nM T00820 CDT8Y9 10185064 EC50 = 1621.81 nM T00820 CN0BY8 10185759 EC50 = 9549.93 nM T00820 CY4F9Q 10203855 EC50 = 2290.87 nM T00820 C0FK5C 10204578 EC50 = 9772.37 nM T00820 CV5PH2 10206849 EC50 = 6760.83 nM T00820 C4Q6IU 10227985 EC50 = 8912.51 nM T00820 CRCH64 10228399 EC50 = 5011.87 nM T00820 C0IG2S 10249251 EC50 = 213 nM T00820 C1JE7N 10254651 EC50 > 10000 nM T00820 CFI14T 10275180 EC50 = 12022.64 nM T00820 CPX05L 10296978 EC50 = 912.01 nM T00820 C9IC3O 10297235 EC50 = 5370.32 nM T00820 C25BIV 10297236 EC50 = 1513.56 nM T00820 CZ9SG4 10298234 EC50 = 1659.59 nM T00820 C29ESL 10298327 EC50 = 1096.48 nM T00820 CEG10L 10318275 EC50 = 46 nM T00820 C2MZ6B 10321166 EC50 = 185 nM T00820 C6SC3D 10321411 EC50 = 98 nM T00820 C8AGW4 10322433 EC50 > 10000 nM T00820 CX96ZS 10341099 EC50 = 9 nM T00820 C6VW2M 10341325 EC50 > 10000 nM T00820 CJSD81 10341635 EC50 = 44 nM T00820 C0I8GP 10342450 EC50 = 76 nM T00820 CHMY27 10345145 EC50 = 306 nM T00820 CW0HA2 10345523 EC50 = 47 nM T00820 CZ2XF0 10362210 EC50 = 751 nM T00820 C4R7VE 10365187 EC50 = 23 nM T00820 CNXC07 10387338 EC50 = 12 nM T00820 CQ28DJ 10408241 EC50 = 177000 nM T00820 C7HBC1 10411024 EC50 = 1750 nM T00820 C51IOT 10411358 EC50 = 2040 nM T00820 C19XMR 10412158 EC50 = 317 nM T00820 COT06Y 10431921 EC50 = 60 nM T00820 C2LOK7 10433766 EC50 = 570 nM T00820 CB2Y3G 10451456 EC50 = 15 nM T00820 C9P8SX 10452297 EC50 = 6630 nM T00820 CVI3A7 10455786 EC50 = 12 nM T00820 CB7AQ8 10456839 EC50 = 117 nM T00820 CUHO58 10458527 EC50 > 10000 nM T00820 C67ZYJ 10459906 EC50 = 154 nM T00820 CX8Q7G 10476467 EC50 = 49 nM T00820 C6BTD9 10477834 EC50 = 70 nM T00820 C6LF4Q 10477835 EC50 = 44 nM T00820 CR2NL6 11742811 EC50 = 81 nM T00820 CB05KW 11754927 EC50 = 160 nM T00820 C9PEL4 23729615 EC50 = 758.58 nM T00820 CU29XL 23729616 EC50 = 2238.72 nM T00820 CW9GN6 23729617 EC50 = 10471.29 nM T00820 CSC6N9 23729618 EC50 = 891.25 nM T00820 CDI1X8 23729711 EC50 = 5370.32 nM T00820 C34SEU 23729712 EC50 = 1737.8 nM T00820 CSGX18 23729713 EC50 = 2570.4 nM T00820 CG5K8O 23729714 EC50 = 2290.87 nM T00820 CXF18B 23729715 EC50 = 3801.89 nM T00820 C4BJ0W 23729716 EC50 = 7762.47 nM T00820 CQ2M1H 23729814 EC50 < 100000 nM T00820 CJ1AY4 23729815 EC50 = 954.99 nM T00820 C5WQS9 23729816 EC50 = 1096.48 nM T00820 CJ5N3K 23729817 EC50 = 1288.25 nM T00820 CHX62L 23729818 EC50 = 2630.27 nM T00820 C23HWA 23729819 EC50 = 2041.74 nM T00820 CBO9F0 23729927 EC50 = 4570.88 nM T00820 C2JF6V 23729928 EC50 = 4265.8 nM T00820 C2WU9I 23729929 EC50 = 4265.8 nM T00820 C4VCF6 23729930 EC50 = 11748.98 nM T00820 CN4IU0 23730737 EC50 = 645.65 nM T00820 CF3G9B 23730848 EC50 = 2041.74 nM T00820 CCD7X5 23730850 EC50 = 2089.3 nM T00820 C0B5OE 23730851 EC50 = 3715.35 nM T00820 CTJ54I 23730852 EC50 = 26915.35 nM T00820 CZ8OS3 23730853 EC50 = 776.25 nM T00820 CKA52B 23730965 EC50 = 1318.26 nM T00820 CQ0C1K 23730966 EC50 = 1659.59 nM T00820 C65EOP 23730967 EC50 < 100000 nM T00820 CTL7N4 23730968 EC50 = 4265.8 nM T00820 COU81D 23730969 EC50 = 8912.51 nM T00820 CUH08M 44293467 EC50 = 4840 nM T00820 CE5SH1 44293670 EC50 = 24 nM T00820 CED32T 44293814 EC50 = 417 nM T00820 CF25KZ 44293901 EC50 = 1160 nM T00820 C93EKW 44436328 EC50 = 338.84 nM T00820 C7HD3B 44436351 EC50 = 1071.52 nM T00820 C9LBX0 44436355 EC50 = 6606.93 nM T00820 CXI5V1 56643481 IC50 > 5000 nM T00820 CH3BN6 56643486 IC50 > 5000 nM T00820 C6XI4W 56647652 IC50 > 5000 nM T00820 CQ0F3N 70693564 EC50 = 2137.96 nM T01282 CKO4M6 56663319 Ki = 68 nM T01282 CY34VE 56677007 Ki = 53 nM T01282 D07ZRG 46899577 Ki = 20 nM T92517 D03ZOR 73356676 IC50 > 1000 nM T92517 D05LZV 71679021 IC50 = 50 nM T92517 D0HZ1Z 71679189 IC50 = 100 nM T92517 D0KA3L 71817936 IC50 = 2500 nM T92517 D0WS4U 71818387 IC50 > 1000 nM T92517 D06VTU 9885817 IC50 = 22 nM T92517 D0G5ZE 72430 Ki = 8 nM T92517 D0NJ1A 65663 IC50 = 4000 nM T92517 CAX1O8 73364 IC50 = 5 nM T92517 CHUX81 121855 IC50 = 23 nM T92517 CK84SO 123664 IC50 = 40 nM T92517 C6J4GA 446403 Ki = 3.4 nM T92517 C3P5YW 456427 IC50 = 8 nM T92517 CWU18B 3082865 IC50 = 33 nM T92517 CK4X9E 5353866 Ki = 260 nM T92517 CNY2T4 6857712 IC50 = 170 nM T92517 CSZ6C3 6918776 IC50 = 13340 nM T92517 CK3Q0Z 6993120 IC50 = 11 nM T92517 CPO9V3 9798553 IC50 = 86 nM T92517 CLTO67 9821317 IC50 > 10000 nM T92517 CCD1U8 9827198 IC50 = 21 nM T92517 C8W9ER 9827472 Ki = 140 nM T92517 C3ZMF4 9828813 IC50 = 50 nM T92517 C42ZQE 9828874 IC50 = 6 nM T92517 CH3D9B 9829045 IC50 = 21 nM T92517 CK2Z4X 9831066 IC50 = 17 nM T92517 CZ3MO5 9839500 Ki = 210 nM T92517 COAM65 9844151 Ki = 8 nM T92517 CH2TD6 9844274 IC50 = 5 nM T92517 C2VX4Z 9848148 Ki = 56 nM T92517 C59TMI 9849265 IC50 = 26 nM T92517 C6SWE8 9868097 IC50 = 7 nM T92517 C6Z4WX 9868717 Ki = 30 nM T92517 CA54DZ 9869293 IC50 = 10 nM T92517 CCA4P9 9869913 IC50 = 19 nM T92517 C3LD8C 9887542 IC50 = 240 nM T92517 C7M0IP 9888995 IC50 = 50 nM T92517 CU01RT 9889401 Ki = 36 nM T92517 C9W3FE 9891793 IC50 = 56 nM T92517 C8WZ6Y 9892354 Ki = 41000 nM T92517 CC8O9R 9915617 IC50 = 28 nM T92517 CG8M2O 9916329 IC50 = 20 nM T92517 C4WDY5 9955551 IC50 = 193 nM T92517 CHA6S8 9956417 IC50 = 21 nM T92517 CLX02R 9960930 IC50 = 17 nM T92517 CF5W3H 9984343 Ki = 2 nM T92517 CR4L2X 9997899 IC50 = 4 nM T92517 C4DF7N 10046879 Ki = 15 nM T92517 C5X2TU 10069167 Ki = 13.3 nM T92517 C4FT1W 10071237 IC50 = 6 nM T92517 C6EHG9 10077274 Ki = 14 nM T92517 CR1NC5 10138215 IC50 = 82 nM T92517 C35QPL 10181824 IC50 = 22.5 nM T92517 CV0CI4 10216098 IC50 = 10 nM T92517 C8IXH2 10252431 IC50 = 25 nM T92517 CTU29C 10254187 IC50 = 370 nM T92517 CFD8Y4 10308902 IC50 = 29 nM T92517 CMR75W 10318568 IC50 = 120 nM T92517 C78XZT 10341806 IC50 = 30 nM T92517 CP1ZM5 10349334 Ki = 8 nM T92517 C7D9XB 10363069 IC50 = 500 nM T92517 CDY26B 10366413 Ki = 6 nM T92517 C31QWD 10376483 IC50 = 1200 nM T92517 C64MUQ 10407439 IC50 = 600 nM T92517 C39LPB 10408446 IC50 = 230 nM T92517 C9IJ6Y 10408700 IC50 = 14 nM T92517 CXL4O2 10457121 Ki = 9 nM T92517 C0Z4IV 10462403 Ki = 14 nM T92517 CO5D0G 10473315 IC50 = 800 nM T92517 C86THD 10600514 Ki = 9 nM T92517 CI4RH6 10623515 Ki = 11 nM T92517 CN8PB5 10649378 Ki = 4 nM T92517 CKGY04 10666857 Ki = 66 nM T92517 CQPW92 10668944 Ki = 41 nM T92517 C0O6PE 10689874 Ki = 9 nM T92517 C3VCM6 10690823 Ki = 11 nM T92517 C0LEN3 10695520 Ki = 22 nM T92517 C0GHV1 10739025 Ki = 28 nM T92517 C0XE7T 10740734 Ki = 9 nM T92517 C5GD2S 10746284 Ki = 19000 nM T92517 C6FVU3 10759604 Ki = 29 nM T92517 CPC98S 10783485 Ki = 36 nM T92517 C5SN8Q 10786038 Ki = 11 nM T92517 CCD76F 10787888 Ki = 10 nM T92517 CD72KH 10788273 Ki = 6 nM T92517 CBK06L 10861643 IC50 = 7.5 nM T92517 CLN9A1 10873870 IC50 = 15 nM T92517 C78SVF 10882836 IC50 = 83 nM T92517 C80GNZ 10884980 IC50 = 30 nM T92517 C5X3RN 10947229 IC50 ~ 5000 nM T92517 C1RTF4 10972257 IC50 = 8 nM T92517 CN1L8Q 10982880 IC50 = 24 nM T92517 C6FN2G 10993481 IC50 = 2200 nM T92517 CN95GJ 11026092 IC50 = 28 nM T92517 CETV63 11036797 IC50 = 37 nM T92517 C23BUM 11122265 IC50 = 1000000 nM T92517 CZV86B 11143626 IC50 = 2400 nM T92517 CN0F8E 11199915 Ki = 10 nM T92517 CFOV37 11237019 IC50 > 1000000 nM T92517 CM8O6L 11257152 IC50 > 100000 nM T92517 CGS8M0 11293792 IC50 = 110 nM T92517 CCV6T0 11374367 IC50 ~ 5000 nM T92517 CHGO82 11406291 IC50 = 40 nM T92517 C3X7AL 11432299 IC50 > 1000000 nM T92517 C4YAB5 11501216 IC50 = 600 nM T92517 C6W5DY 11559647 IC50 = 180 nM T92517 CI8N7S 11574155 IC50 = 150 nM T92517 C5OBL4 11609750 IC50 = 630 nM T92517 C3UC2D 11617861 IC50 = 220 nM T92517 COV96I 11646523 IC50 = 140 nM T92517 C7CL1E 11660607 IC50 = 240 nM T92517 CTQC50 11682173 IC50 = 150 nM T92517 C1C2NQ 11717569 IC50 = 910 nM T92517 C7V8PD 11717773 IC50 = 260 nM T92517 CB5Y1Z 11796288 Ki = 370 nM T92517 CY2R8A 11797679 IC50 = 56 nM T92517 CVBX10 11824872 IC50 = 14000 nM T92517 C6OYI8 11825185 IC50 = 130 nM T92517 CZI24R 12039099 IC50 = 700 nM T92517 C3RYT7 13388085 Ki = 1080 nM T92517 CG2H0I 13696522 IC50 = 10000 nM T92517 CCQ07Z 15168140 IC50 = 500 nM T92517 CTA73X 15168141 IC50 = 300 nM T92517 C21ZHN 15168142 IC50 = 1000 nM T92517 C65HMZ 15168143 IC50 = 6000 nM T92517 CMK53T 15168144 IC50 = 2000 nM T92517 CNRX46 15168145 IC50 = 1000 nM T92517 CS35MQ 15168146 IC50 = 5000 nM T92517 CT7D8X 15168147 IC50 = 2000 nM T92517 C41AJC 15168153 IC50 = 4000 nM T92517 C5MX1W 15838740 Ki = 810 nM T92517 CM56TF 16127556 IC50 = 3 nM T92517 CUA19Y 16760339 Ki = 250 nM T92517 CYA5V6 16760340 Ki = 19 nM T92517 C3P1ZQ 18458068 IC50 = 130 nM T92517 C9NB3C 18691001 Ki = 40 nM T92517 COG43Z 18691004 Ki = 80 nM T92517 CF89DV 18734983 Ki = 460 nM T92517 C0M5DN 18734989 Ki = 33000 nM T92517 C7ER8G 19959063 IC50 = 7000 nM T92517 C2GOC5 19959066 IC50 = 5000 nM T92517 CLM2E4 19959068 IC50 = 2000 nM T92517 CS5NM0 19959069 IC50 = 500 nM T92517 C6E8KW 19959071 IC50 = 10000 nM T92517 CO7F9J 19959072 IC50 = 2000 nM T92517 CWT94S 19959085 IC50 = 20000 nM T92517 CBR2I6 19959088 IC50 = 2000 nM T92517 CJ9I5P 20666711 Ki = 280 nM T92517 C2BEJ1 20666712 Ki = 140 nM T92517 CQ7W4F 21190792 Ki = 450 nM T92517 C4HNB1 21190800 Ki = 90 nM T92517 CZL02V 21190806 Ki = 450 nM T92517 CZ8L3Q 21190807 Ki = 230 nM T92517 CFL9G6 21190822 Ki = 40 nM T92517 C28QTJ 21190825 Ki = 50 nM T92517 CY06OB 21190844 Ki = 50 nM T92517 C0VJ9Z 21190850 Ki = 200 nM T92517 CXU73K 21190899 Ki = 370 nM T92517 CI57HS 22988111 Ki = 125 nM T92517 CJD86W 23240735 Ki = 680 nM T92517 C6YW0C 23240737 Ki = 200 nM T92517 C15TFI 23240738 Ki = 200 nM T92517 C2NRA7 23240739 Ki = 52 nM T92517 C6YRN8 24822372 IC50 = 190 nM T92517 CQYO68 24822373 IC50 = 220 nM T92517 CH4Z5E 24822532 IC50 = 420 nM T92517 C75PMR 24936064 IC50 = 710 nM T92517 CGQC69 25013878 IC50 > 30000 nM T92517 CJV8E7 25156794 Ki = 21 nM T92517 C7BR6I 25157065 Ki = 38 nM T92517 CRT89B 25157358 Ki = 32 nM T92517 CJ9QZ6 25157359 Ki = 20 nM T92517 CQ6UX0 25157961 Ki = 45 nM T92517 CAC2G6 42597070 IC50 = 2810 nM T92517 CW8BM0 42597071 IC50 = 40170 nM T92517 CP0GO6 42597072 IC50 = 6190 nM T92517 CGU46I 42597073 IC50 = 22130 nM T92517 CN6UZ9 42597074 IC50 = 7410 nM T92517 C9AID4 42597314 IC50 = 34010 nM T92517 CMH05R 42600221 IC50 = 91420 nM T92517 CEQ5L8 42600222 IC50 > 100000 nM T92517 CV7EU3 42600223 IC50 = 64610 nM T92517 CIRO21 42600463 IC50 = 35260 nM T92517 C8PC3T 42600464 IC50 = 84750 nM T92517 CF6O0H 42600465 IC50 = 6190 nM T92517 C8Y9NQ 44219712 IC50 = 3170 nM T92517 C37AEK 44265286 IC50 = 5 nM T92517 CM52WS 44265321 IC50 = 56 nM T92517 CZ4E9D 44265330 IC50 = 50 nM T92517 CJ0FL3 44265335 IC50 = 47 nM T92517 CWY67K 44265357 IC50 = 240 nM T92517 CRE64F 44265358 IC50 = 170 nM T92517 CR9Z8F 44265359 IC50 = 195 nM T92517 CITB32 44265381 IC50 = 76 nM T92517 CY1C9F 44265390 IC50 = 200 nM T92517 C0K7YW 44265402 IC50 = 1000 nM T92517 CV54IT 44265411 IC50 = 1000 nM T92517 C6OQT7 44265417 IC50 = 81 nM T92517 CK7HP0 44265418 IC50 = 7 nM T92517 CG4D1L 44265420 IC50 = 205 nM T92517 CE5Q8Y 44265428 IC50 = 286 nM T92517 CO19RW 44265429 IC50 = 20 nM T92517 C96SLN 44265434 IC50 = 20 nM T92517 C9L6WF 44265439 IC50 = 500 nM T92517 CLK2T1 44265440 IC50 = 5000 nM T92517 CU13OY 44265441 IC50 = 200 nM T92517 C86SBG 44265442 IC50 = 63 nM T92517 C0K5JY 44265443 IC50 = 155 nM T92517 C5C7KM 44265444 IC50 = 150 nM T92517 CA7MO2 44265449 IC50 = 2400 nM T92517 CK3MN8 44265450 IC50 = 29 nM T92517 CK35CW 44265451 IC50 = 56 nM T92517 CY6HT7 44265455 IC50 = 35 nM T92517 CO37LC 44265456 IC50 = 5000 nM T92517 C6UHC7 44265457 IC50 = 340 nM T92517 CYD70I 44265462 IC50 = 89 nM T92517 CBC4P5 44288507 IC50 = 138 nM T92517 CH4OQ7 44288508 IC50 = 130 nM T92517 C19RJI 44288910 IC50 = 50 nM T92517 CBO9Y1 44304780 IC50 = 2000 nM T92517 CWSK27 44304781 IC50 = 100000 nM T92517 COX2J1 44309545 Ki = 560 nM T92517 CYS85H 44309591 Ki = 160 nM T92517 CZ50QH 44309592 Ki = 1350 nM T92517 C4GVT2 44309610 Ki = 670 nM T92517 CDNF42 44309623 Ki = 13500 nM T92517 CD6O5C 44309624 Ki = 13600 nM T92517 CNCM35 44309687 Ki = 800000 nM T92517 C7TR9Z 44309707 Ki = 450 nM T92517 C0JPT5 44309797 Ki = 960 nM T92517 CTF98D 44315377 Ki = 56000 nM T92517 CFM96P 44315648 Ki = 2000 nM T92517 CO4C9E 44315766 Ki = 33 nM T92517 CDY5W6 44315767 Ki = 400 nM T92517 CL1VN6 44315859 Ki = 21 nM T92517 CNY81T 44315869 Ki = 420 nM T92517 CO8L1W 44315978 Ki = 10 nM T92517 CTVR80 44315979 Ki = 71 nM T92517 C90SRY 44316019 Ki ~ 360 nM T92517 CIRD94 44316029 Ki = 130 nM T92517 CK5XY6 44316030 Ki = 15 nM T92517 CP8WY4 44316032 Ki = 59 nM T92517 CP86JI 44316033 Ki = 570 nM T92517 C28FXM 44316100 Ki = 400 nM T92517 C1MU5L 44316138 Ki = 430 nM T92517 C28IJA 44316139 Ki = 46 nM T92517 CV2OZ3 44316148 Ki = 26 nM T92517 C8XE3U 44316174 Ki = 21 nM T92517 C46JHA 44316175 Ki = 1100 nM T92517 CBG3Z4 44316227 Ki = 49 nM T92517 CRC1B6 44316228 Ki = 130 nM T92517 C7J6ZK 44316248 Ki = 1100 nM T92517 C8GQM6 44316295 Ki = 62 nM T92517 C8DQ1J 44316385 Ki > 1000 nM T92517 CCWR05 44316386 Ki = 57 nM T92517 CXDI94 44317334 Ki = 27 nM T92517 CNBR62 44317343 Ki = 18.3 nM T92517 CS23PT 44317344 Ki = 15 nM T92517 CV23BP 44317348 Ki = 8.4 nM T92517 C09WVA 44321581 IC50 = 12 nM T92517 C6LH3B 44321603 IC50 = 152 nM T92517 CA56UP 44321953 IC50 = 28 nM T92517 C8DX6O 44322591 IC50 = 45 nM T92517 CV2C4T 44322992 IC50 = 53 nM T92517 C0PV5A 44323013 IC50 = 125 nM T92517 CP2IG8 44323050 IC50 = 13 nM T92517 C3KU0G 44323051 IC50 = 41 nM T92517 C5OT0F 44323240 Ki = 9 nM T92517 C94FID 44330054 IC50 = 500 nM T92517 C5CSJ7 44330064 IC50 = 75 nM T92517 CC1W7N 44330831 Ki = 93 nM T92517 CZ65KO 44330832 Ki > 1500 nM T92517 CA30IY 44330865 Ki = 61 nM T92517 C9VL8D 44330887 Ki = 333 nM T92517 CMX96T 44330903 Ki = 66 nM T92517 C9Y7KD 44330914 Ki = 32 nM T92517 CUM39I 44330915 Ki = 74 nM T92517 C5M7NT 44330942 Ki = 129 nM T92517 CSD1Q3 44330943 Ki = 170 nM T92517 CPNJ80 44330944 Ki = 77 nM T92517 CK4MB6 44330965 Ki = 244 nM T92517 C0MS7A 44330966 Ki = 116 nM T92517 CBFT17 44330977 Ki = 119 nM T92517 CX3OE2 44330979 Ki > 350000 nM T92517 C5AN6S 44330981 Ki = 718 nM T92517 CN4HM2 44330982 Ki = 92 nM T92517 C8C4MB 44342381 IC50 = 28 nM T92517 CN5GQ3 44343531 Ki = 350 nM T92517 CGN37W 44343594 Ki = 800 nM T92517 C47KQO 44343612 Ki = 200 nM T92517 C56PAB 44344207 IC50 = 28 nM T92517 CBS68D 44344211 IC50 = 85 nM T92517 CJF12T 44344229 IC50 = 150 nM T92517 C2X4VC 44344230 IC50 = 38 nM T92517 CU5V3I 44344296 IC50 = 37 nM T92517 C4JS8H 44344344 IC50 = 30 nM T92517 CQG1N0 44344349 IC50 = 36 nM T92517 CXC5E2 44344363 IC50 = 200 nM T92517 CS6E0V 44344391 IC50 = 7 nM T92517 C1XUF0 44344531 IC50 = 11 nM T92517 CHP35Z 44349441 IC50 = 147 nM T92517 C1MY4C 44349727 IC50 = 20 nM T92517 C5N1JX 44350690 IC50 = 6000 nM T92517 CIJ38P 44350713 IC50 = 430 nM T92517 CQ2S5A 44350722 IC50 = 370 nM T92517 CZAY62 44350724 IC50 > 10000 nM T92517 CD0FW8 44350732 IC50 = 5200 nM T92517 CR6K8M 44350733 IC50 = 7 nM T92517 CNM89X 44350737 IC50 > 10000 nM T92517 CXQ98I 44350761 IC50 = 350 nM T92517 CCR71B 44350770 IC50 = 7400 nM T92517 CWZC60 44350771 IC50 = 600 nM T92517 C5O1IV 44350776 IC50 > 10000 nM T92517 CW5GU7 44350932 IC50 = 30000 nM T92517 C4L6EC 44350965 IC50 = 20000 nM T92517 CXID91 44350996 IC50 = 2000 nM T92517 C93RZA 44351015 IC50 = 2000 nM T92517 CS8F0V 44351163 IC50 = 30000 nM T92517 C6X9JO 44353497 Ki = 350 nM T92517 CVHL49 44353498 Ki = 500 nM T92517 C50JMZ 44353509 Ki = 7900 nM T92517 C1R7HO 44353510 Ki = 1400 nM T92517 CD1KB5 44353514 Ki = 7800 nM T92517 CT43EV 44353526 Ki = 850 nM T92517 CV6U1K 44353527 Ki = 250 nM T92517 CN15EA 44353530 Ki = 280 nM T92517 CKH5Y4 44353532 Ki = 460 nM T92517 CK35CO 44353533 Ki = 700 nM T92517 CUFZ01 44353534 Ki = 620 nM T92517 CN6B8M 44353535 Ki = 1300 nM T92517 C0T4MF 44353540 Ki = 1300 nM T92517 CP5NY3 44353544 Ki = 160 nM T92517 CB1HC7 44353545 Ki = 750 nM T92517 C5FXE6 44353552 Ki = 290 nM T92517 CH3BQ1 44353553 Ki = 5000 nM T92517 CJ0Y3M 44353556 Ki = 1000 nM T92517 C1QG3Z 44353580 Ki = 120 nM T92517 C6T3DA 44353581 Ki = 110 nM T92517 CV6U5Q 44353582 Ki = 130 nM T92517 CMTJ91 44353589 Ki = 300 nM T92517 CM3R5T 44353590 Ki = 650 nM T92517 CZ2YG8 44353593 Ki = 410 nM T92517 CFZ36E 44353603 Ki = 220 nM T92517 C6MV2C 44353604 Ki = 120 nM T92517 CWV2C8 44353606 Ki = 200 nM T92517 CEJ3D8 44353608 Ki = 1100 nM T92517 C8YPO1 44353613 Ki = 380 nM T92517 C0WIP1 44353630 Ki = 1100 nM T92517 CT3Q8G 44353631 Ki = 10000 nM T92517 C6BQS9 44353632 Ki = 800 nM T92517 C7DRX0 44353633 Ki = 500 nM T92517 C0T5HM 44353640 Ki = 1900 nM T92517 CS9VG4 44353649 Ki = 800 nM T92517 CI9UB0 44353680 Ki = 230 nM T92517 C1V8RS 44353769 Ki = 640 nM T92517 C1ATV5 44353779 Ki = 240 nM T92517 C53QGD 44353782 Ki = 330 nM T92517 C91OHB 44353783 Ki = 800 nM T92517 CUY2N7 44353792 Ki = 650 nM T92517 C5XVK9 44353793 Ki = 2300 nM T92517 CTD5O8 44353799 Ki = 350 nM T92517 CH80QO 44353801 Ki = 420 nM T92517 CNM2U3 44353805 Ki = 650 nM T92517 CF8ZU0 44353806 Ki = 32000 nM T92517 CV97ZN 44353808 Ki = 100 nM T92517 CG6Q3F 44353809 Ki = 900 nM T92517 C8O3LK 44353810 Ki = 350 nM T92517 CMP1Z0 44353811 Ki = 50 nM T92517 CPA90D 44353812 Ki = 250 nM T92517 C49MCW 44353814 Ki = 130 nM T92517 CN9W5C 44353816 Ki = 200 nM T92517 CX3RZ0 44353817 Ki = 200 nM T92517 CCEU50 44353818 Ki = 500 nM T92517 C57SFJ 44353819 Ki = 480 nM T92517 CX9LJ0 44353820 Ki = 590 nM T92517 C9PY1J 44353821 Ki = 180 nM T92517 CU74GM 44353822 Ki = 350 nM T92517 CDHX90 44353823 Ki = 120 nM T92517 CQ9BT7 44353833 Ki = 330 nM T92517 CT21FG 44353834 Ki = 380 nM T92517 CZ3XP9 44353836 Ki = 300 nM T92517 CB7I6Q 44353838 Ki = 600 nM T92517 CB7P0H 44353839 Ki = 760 nM T92517 CF3A0M 44353840 Ki = 70 nM T92517 CS5DX4 44353841 Ki = 80 nM T92517 CZ89JO 44353846 Ki = 500 nM T92517 CP3VT2 44353858 Ki = 1200 nM T92517 C5H9VR 44353859 Ki = 110 nM T92517 C1HR8U 44353865 Ki = 270 nM T92517 C19QIH 44366718 IC50 > 10000 nM T92517 CWY6G7 44366744 IC50 = 35 nM T92517 C8CA9M 44366904 IC50 = 35 nM T92517 C09UJA 44366905 IC50 > 1000 nM T92517 CHOA20 44366907 IC50 >> 10000 nM T92517 CZF16C 44366908 IC50 = 41 nM T92517 CO3AW0 44366909 IC50 = 580 nM T92517 CPKD86 44366920 IC50 = 120 nM T92517 CSQ5G7 44366942 IC50 = 370 nM T92517 CO92LE 44366950 IC50 = 18 nM T92517 CU65DO 44366951 IC50 >> 10000 nM T92517 C7BSI0 44366966 IC50 = 140 nM T92517 CE4LP6 44366970 IC50 > 1000 nM T92517 COVY42 44366975 IC50 = 33 nM T92517 C6B4PU 44366976 IC50 = 530 nM T92517 C6YLJ4 44366977 IC50 = 120 nM T92517 C8CVW5 44366981 IC50 = 190 nM T92517 CU1O7M 44366983 IC50 = 4 nM T92517 C68VQF 44367018 IC50 > 1000 nM T92517 C7O0SF 44367033 IC50 = 8 nM T92517 C9GTP7 44367043 IC50 = 10 nM T92517 CPIA97 44367088 IC50 = 5 nM T92517 CT8V0P 44367090 IC50 ~ 10000 nM T92517 CY2S7M 44367093 IC50 = 7 nM T92517 C96JGV 44367108 IC50 = 37 nM T92517 CRO6B5 44367143 IC50 > 1000 nM T92517 CI06PV 44367144 IC50 = 15 nM T92517 CCJ82Q 44367145 IC50 = 300 nM T92517 C0R8XB 44367146 IC50 = 11 nM T92517 CRJ60P 44367166 IC50 = 33 nM T92517 C9HVD2 44367167 IC50 = 62 nM T92517 C20ZEX 44367168 IC50 ~ 1000 nM T92517 C2GXL4 44367194 IC50 = 45 nM T92517 C1P7BN 44367195 IC50 = 17 nM T92517 C2P9AV 44367196 IC50 = 6 nM T92517 C4BGE1 44367197 IC50 = 72 nM T92517 CH4R3S 44367198 IC50 = 110 nM T92517 CDK27F 44367200 IC50 = 150 nM T92517 CEC27U 44367201 IC50 = 32 nM T92517 CSM2K6 44367211 IC50 = 31 nM T92517 CC08ZH 44367212 IC50 = 12 nM T92517 C02RLM 44367214 IC50 = 20 nM T92517 C0T2SB 44367215 IC50 = 12 nM T92517 CL6YN0 44367223 IC50 ~ 10000 nM T92517 CAG85M 44367224 IC50 = 11 nM T92517 CVE1D6 44367230 IC50 = 25 nM T92517 C6R9ZP 44367238 IC50 = 12 nM T92517 C82NVJ 44367239 IC50 = 11 nM T92517 C9M2KI 44367242 IC50 = 19 nM T92517 C1QV7T 44367278 IC50 = 15 nM T92517 CC67DA 44367279 IC50 ~ 10000 nM T92517 CJ0Q8N 44367283 IC50 = 10 nM T92517 CC8VU9 44367288 IC50 = 68 nM T92517 C9QS7J 44367294 IC50 = 1200 nM T92517 C09HOB 44367295 IC50 = 90 nM T92517 C5FD6A 44367313 IC50 = 8 nM T92517 C8U7KZ 44367330 IC50 = 1100 nM T92517 CGB4V7 44367332 IC50 = 15 nM T92517 C7HMZ4 44367334 IC50 = 40 nM T92517 CAPG41 44381683 IC50 = 27 nM T92517 CY68TS 44381691 IC50 = 10 nM T92517 CJ69ZD 44381692 IC50 = 630 nM T92517 C4AZS8 44381725 IC50 = 130 nM T92517 CLVI37 44381726 IC50 = 18 nM T92517 C5LK6Y 44381744 IC50 = 13 nM T92517 CGXL04 44381745 IC50 = 31 nM T92517 CTB1X4 44381873 IC50 = 28 nM T92517 C3XJI4 44381886 IC50 = 830 nM T92517 CG49KD 44381888 IC50 = 260 nM T92517 CHF32N 44381900 IC50 = 14 nM T92517 CK05YD 44381932 IC50 = 21000 nM T92517 C4AF9C 44381950 IC50 = 23 nM T92517 CRO09I 44381951 IC50 = 14 nM T92517 CZF10N 44402392 IC50 = 2480 nM T92517 CP9H7I 44402434 IC50 = 450 nM T92517 C1S8ZC 44402519 IC50 = 8170 nM T92517 C7MGX5 44402520 IC50 > 20000 nM T92517 C5ZMY7 44402533 IC50 = 720 nM T92517 CFY74K 44402562 IC50 = 810 nM T92517 CATR89 44402636 IC50 = 530 nM T92517 C71JRQ 44402637 IC50 = 4530 nM T92517 CJW7N1 44402655 IC50 = 8730 nM T92517 CBAM59 44402720 IC50 = 5690 nM T92517 CG42KX 44402844 IC50 > 20000 nM T92517 C3AYM7 44412929 IC50 > 100000 nM T92517 C8YR5A 44413024 IC50 = 880 nM T92517 C9FIN7 44446395 IC50 = 8620 nM T92517 CK0IC6 44446396 IC50 = 40170 nM T92517 C0ETX2 44446397 IC50 > 50000 nM T92517 CA4OU8 44446398 IC50 = 5010 nM T92517 CI4G2Q 44446399 IC50 = 3810 nM T92517 C5W4PS 44446400 IC50 = 1780 nM T92517 C6MU5N 44446401 IC50 = 5630 nM T92517 C25KUT 44446402 IC50 = 7720 nM T92517 C34SHV 44446403 IC50 = 3710 nM T92517 CSAW74 44446404 IC50 = 730 nM T92517 CMJ0O1 44446405 IC50 = 6280 nM T92517 CLH74F 44565900 IC50 = 1690 nM T92517 CMIP10 44565901 IC50 = 3530 nM T92517 CU54ZD 44565902 IC50 > 30000 nM T92517 CX3D7I 44565903 IC50 > 30000 nM T92517 CHBZ57 44565904 IC50 > 30000 nM T92517 CP5S2B 44565923 IC50 > 30000 nM T92517 CY5XC6 44565924 IC50 > 30000 nM T92517 C70BXJ 44565925 IC50 = 277 nM T92517 CW8A7S 44565926 IC50 > 30000 nM T92517 CG5R1M 44565927 IC50 > 30000 nM T92517 CB6F4H 44565978 IC50 > 30000 nM T92517 C2LC5N 44565979 IC50 > 30000 nM T92517 CS6YO0 44566187 IC50 = 4560 nM T92517 CSF17Z 44566188 IC50 = 7430 nM T92517 CH5WK2 44566189 IC50 > 30000 nM T92517 CESA78 44566194 IC50 > 30000 nM T92517 CJP3U5 44566195 IC50 = 2390 nM T92517 CUFJ57 44566196 IC50 = 3160 nM T92517 CGP6X5 44566197 IC50 = 19200 nM T92517 CJ35AL 44566198 IC50 > 30000 nM T92517 C5YQP1 44581192 IC50 = 6250 nM T92517 CR5H0E 44581193 IC50 = 3200 nM T92517 CBW4Z6 44581194 IC50 = 3330 nM T92517 CI0PQ8 44581195 IC50 = 540 nM T92517 C25OEA 44581234 IC50 = 4290 nM T92517 C80BVR 44581282 IC50 = 340 nM T92517 CTS0E2 44581283 IC50 = 13840 nM T92517 C4CQ7G 44581284 IC50 = 6160 nM T92517 CCW53D 44581285 IC50 = 1180 nM T92517 CI56KU 44581319 IC50 = 4250 nM T92517 C0N7HI 44581320 IC50 = 700 nM T92517 CZ2R4O 44581321 IC50 = 5730 nM T92517 CBP0Y7 44581322 IC50 = 3770 nM T92517 C1IO0W 44581360 IC50 = 520 nM T92517 C7EWP0 44581387 IC50 = 2350 nM T92517 CRL91Q 44581388 IC50 = 1640 nM T92517 CV6ML0 44581389 IC50 = 2090 nM T92517 CASI41 44581412 IC50 = 950 nM T92517 C57VEF 44581413 IC50 = 2130 nM T92517 C0Q6XJ 44581414 IC50 = 8000 nM T92517 C0CLO7 44581415 IC50 = 1860 nM T92517 CSL40T 44581416 IC50 = 12990 nM T92517 CXN5S2 46861589 Ki = 38 nM T92517 C8T5BF 46870403 Ki = 234 nM T92517 C7TI9G 46870676 Ki = 82 nM T92517 CN0G3B 46870679 Ki = 177 nM T92517 C1PLT8 46870767 Ki = 122 nM T92517 C7OYW5 46944251 Ki = 36 nM T92517 CT6MR0 49785938 Ki = 82 nM T92517 CUL18R 53245743 Ki = 120 nM T92517 C3FRT7 53245744 Ki = 205 nM T92517 CW4A6Y 53257219 Ki = 75 nM T92517 C67PKG 53257329 Ki = 120 nM T92517 CKC5M7 53257332 Ki = 150 nM T92517 CLHB63 53257442 Ki = 265 nM T92517 CO2F7A 53257443 Ki = 90 nM T92517 C1CTU6 53258927 Ki = 110 nM T92517 C3OHD0 53258928 Ki = 185 nM T92517 CDQC42 53258931 Ki = 220 nM T92517 CL0O1A 53311527 Ki = 470 nM T92517 CZGD97 53311606 Ki = 490 nM T92517 C8EKO4 53311607 Ki = 480 nM T92517 C0Y3TU 53311694 Ki = 210 nM T92517 CD3C6M 53311695 Ki = 330 nM T92517 CYI3S9 54581933 IC50 = 6070 nM T92517 C8DFA4 54582856 IC50 = 460 nM T92517 C2U5BR 54582857 IC50 = 130 nM T92517 CSM6P7 54582882 IC50 = 670 nM T92517 C53MKE 54582883 IC50 = 320 nM T92517 CQX6V1 54583865 IC50 = 360 nM T92517 C52UXT 54583887 IC50 = 630 nM T92517 CE8XS6 54583888 IC50 = 1380 nM T92517 CK51GA 54585769 IC50 = 610 nM T92517 CPL04M 54587807 IC50 = 500 nM T92517 CDC60L 56675137 IC50 = 1000 nM T92517 C4U2TN 66644532 Ki > 1350 nM T92517 C1KP0Q 66644581 Ki = 125 nM T92517 C2SH6G 66644613 Ki = 528 nM T92517 C29EMR 66644662 Ki = 180 nM T92517 CZ5HL4 66644716 Ki = 268 nM T92517 C13VHL 66644738 Ki = 64 nM T92517 CZN3G2 66644766 Ki = 57 nM T92517 CP5W3K 66644843 Ki = 59 nM T92517 CO48SZ 66644846 Ki = 50 nM T92517 CQS15R 66645094 Ki = 101 nM T92517 CXFR19 66645141 Ki = 90 nM T92517 CJTN62 66719865 Ki = 8 nM T92517 C9WAE4 66719910 Ki = 41 nM T92517 C2U4TJ 66720004 Ki = 100 nM T92517 CBW1U6 66720010 Ki = 690 nM T92517 CE34UA 66720064 Ki = 56 nM T92517 CABJ13 66720066 Ki = 43 nM T92517 C7ES3T 66720071 Ki = 81 nM T92517 C9FQG2 66720098 Ki = 18 nM T92517 CJN72S 66720101 Ki = 72 nM T92517 C8P4KO 66720112 Ki = 88 nM T92517 CNE69H 66720134 Ki = 10 nM T92517 CZO2D6 66720146 Ki = 40 nM T92517 CB4M3Y 66720148 Ki = 83 nM T92517 CZ50KT 66720197 Ki = 34 nM T92517 CKWB70 66720314 Ki = 46 nM T92517 CDA2M1 66995873 Ki = 109 nM T92517 CSF8Z4 67094715 Ki = 73 nM T92517 C90IYL 67094752 Ki = 165 nM T92517 C23OZR 67094880 Ki = 26 nM T92517 CF95AE 67095000 Ki = 39 nM T92517 CK6WL2 67095005 Ki = 110 nM T92517 C4HYT0 67095273 Ki = 48 nM T92517 CB59FX 67095330 Ki = 130 nM T92517 C3ZDV7 67095466 Ki = 70 nM T92517 CUZ68H 67238226 Ki = 380 nM T92517 C3XF5I 67238746 Ki = 550 nM T92517 C08QLD 67239197 Ki = 110 nM T92517 C9DJQ3 71660816 IC50 = 100 nM T92517 CDP98H 71679022 IC50 = 100 nM T92517 CS6G2A 71679023 IC50 = 100 nM T92517 CVOG82 71679190 IC50 = 250 nM T92517 CX9K7L 71768848 Ki = 146 nM T92517 CF04GZ 71817783 IC50 = 100 nM T92517 CM12CF 71817784 IC50 = 150 nM T92517 C1V5SA 71817785 IC50 = 100 nM T92517 CYS6Z5 71817786 IC50 = 100 nM T92517 CA84LP 71817935 IC50 = 5000 nM T92517 CG0BP4 71817937 IC50 = 100 nM T92517 C80HQK 71817939 IC50 = 1000 nM T92517 CA8YK6 71817940 IC50 = 1500 nM T92517 C1S4BQ 71818081 IC50 = 5000 nM T92517 CLGP08 71818082 IC50 = 400 nM T92517 C1RYO3 71818083 IC50 > 1000 nM T92517 CG6C7T 71818084 IC50 > 1000 nM T92517 C5N7HA 71818085 IC50 = 40 nM T92517 CRPX75 71818226 IC50 > 1000 nM T92517 CZRM61 71818227 IC50 > 1000 nM T92517 C65RXL 71818383 IC50 = 300 nM T92517 C8ITL0 73107490 Ki = 310 nM T92517 CE7Z0K 73346021 IC50 = 5000 nM T92517 C36LPI 73346790 IC50 = 100 nM T92517 C2H6BZ 73347050 IC50 = 10 nM T92517 CBES97 73347304 IC50 = 29600 nM T92517 C48HAX 73349081 IC50 > 1000 nM T92517 COF4E6 73349875 IC50 = 28 nM T92517 CMN72X 73352839 IC50 = 28 nM T92517 CS9QO6 73356675 IC50 = 225 nM T92517 CSL0C4 73356677 IC50 = 530 nM T92517 CTA8U5 85090477 Ki = 370 nM T92517 CLJ56E 86647370 Ki = 4360 nM T92517 C2VJ0N 90644780 Ki = 12500 nM T92517 CEZV52 90644781 Ki = 17140 nM T92517 C5E6BQ 90644782 Ki = 21920 nM T92517 C2ZED8 90644783 Ki > 100000 nM T92517 C68OGA 90644784 Ki > 50000 nM T92517 C0CL3K 90644785 Ki = 23730 nM T92517 CQ2RP1 90644786 Ki = 8380 nM T92517 C8EDQ4 90644787 Ki > 100000 nM T92517 CWB19V 90644788 Ki > 100000 nM T92517 C10MVG 90644789 Ki > 100000 nM T92517 C37YFC 90644790 Ki = 3700 nM T92517 C1AR8V 90644791 Ki > 100000 nM T92517 CY0G3V 90644792 Ki > 50000 nM T92517 C2U1KX 90644793 Ki = 30840 nM T92517 C4ANR2 90644794 Ki = 26330 nM T92517 C67WRL 90644795 Ki > 50000 nM T92517 CLMJ40 90644796 Ki > 100000 nM T92517 CQ1F6R 90644797 Ki > 100000 nM T92517 CGQ18K 122197351 Ki = 220 nM T92517 CX7FP8 122197352 Ki = 380 nM T92517 CHJS25 136056122 IC50 = 7000 nM T92517 CD4C1E 136237292 IC50 = 380 nM T92517 CV2P5G 136265721 IC50 = 20 nM T92517 CD95AK 136265747 IC50 = 460 nM T92517 CE0IH1 136265755 IC50 > 1000 nM T92517 C63PBY 136617839 IC50 > 1000 nM T92517 CCT4X0 137645946 Ki = 48 nM T92517 CQJK98 137650664 Ki = 38 nM T92517 CM4ZW3 137651124 Ki = 250 nM T92517 CH18LO 137653371 Ki = 101 nM T92517 CH5G7E 137656944 Ki = 94 nM T92517 CXYK41 137660001 Ki = 164 nM T92517 CE4RZ9 145955916 Ki = 9 nM T92517 C7MVT4 145979463 Ki = 1060 nM T92517 CRW7T5 145980079 IC50 = 1020 nM T92517 C9V5WT 145981454 Ki > 5000 nM T92517 CDXZ97 145981521 Ki = 950 nM T92517 CLF45K 145982180 IC50 = 350 nM T92517 C3CO7L 145982267 IC50 > 1000 nM T92517 CT81XF 145982281 Ki = 2600 nM T92517 CIGY69 145988001 Ki = 1350 nM T92517 CRO2Z8 145988142 IC50 = 1080 nM T92517 CR9O4B 145988599 IC50 > 1000 nM T92517 CE0H1Q 145990917 IC50 > 1000 nM T92517 C9HSN3 155512048 Ki = 200 nM T92517 C0OXS6 155519935 Ki = 240 nM T92517 CM49IT 155523149 Ki = 530 nM T92517 C2MDC3 155525781 Ki = 46 nM T92517 C4I8HO 155533131 Ki = 1350 nM T92517 CT7AC5 155547700 Ki = 545 nM T92517 C0XTM2 155550565 Ki = 9700 nM T92517 C8ELW3 155551211 Ki = 50 nM T92517 CPEZ36 155566005 Ki = 129 nM T92517 D01HUQ 10129992 IC50 = 1400 nM T92517 D03UYO 44353781 Ki = 1100 nM T92517 D06FFP 443118 IC50 > 1000 nM T92517 D08KCA 72429 IC50 = 300 nM T92517 D09FGQ 123985 IC50 = 100 nM T92517 D0Y5IQ 44255320 IC50 = 10000 nM T39195 CO5Y7H 725447 IC50 = 106000 nM T39195 CPJ28H 828532 IC50 = 970 nM T39195 CJ1GN3 869194 IC50 = 101000 nM T39195 CBFT53 975107 IC50 > 30000 nM T39195 CQUP23 2208579 IC50 = 87000 nM T39195 C97ZIP 2262135 IC50 = 99000 nM T39195 C74DMH 2262990 IC50 = 112000 nM T39195 CPR2F8 2931274 IC50 = 96000 nM T39195 CQPJ74 2938648 IC50 = 3430 nM T39195 C6WU4N 5000438 IC50 > 30000 nM T39195 CHY56L 5729350 IC50 = 122000 nM T39195 CI69XU 5739522 IC50 = 108000 nM T39195 CAF89H 25400592 IC50 = 100 nM T39195 CS9TK6 38335241 IC50 = 10300 nM T39195 C78DJQ 71711730 IC50 < 10000 nM T39195 C6RDX4 122192767 Ki = 0.4 nM T39195 CY0K9V 122192770 Ki = 1.2 nM T39195 CDCG19 122192781 Ki = 2 nM T39195 CD5SN7 122192782 Ki = 7 nM T39195 CW9NJ0 134415778 IC50 = 8 nM T39195 CDQ62V 137637214 Ki > 50000 nM T39195 C2K8JV 137639385 Ki = 2000 nM T39195 CNX46H 137654508 Ki > 50000 nM T39195 CUZ35A 138115400 IC50 = 3981.07 nM T39195 CZR36C 155511554 IC50 = 1995.26 nM T39195 C6NX4K 155519661 IC50 = 125.89 nM T39195 C4MS1B 155519676 IC50 = 31622.78 nM T39195 CRC6L7 155524551 Ki = 79 nM T39195 C6L1WU 155525184 Ki = 25 nM T39195 CN3BH5 155527998 IC50 = 398.11 nM T39195 CHYW65 155528639 IC50 = 199.53 nM T39195 CD7O2G 155530095 IC50 = 12589.25 nM T39195 C35QWO 155531023 IC50 = 398.11 nM T39195 CDT7A9 155531797 Ki = 18 nM T39195 C12HON 155536142 IC50 = 12589.25 nM T39195 CY6DK3 155540964 IC50 = 251.19 nM T39195 CU52QS 155545897 Ki > 10000 nM T39195 CH2S6R 155546346 Ki > 10000 nM T39195 C5MB9R 155547962 IC50 = 1584.89 nM T39195 CLFB25 155548371 IC50 = 25118.86 nM T39195 COM52R 155551892 IC50 = 316.23 nM T39195 CJ3FI5 155553630 IC50 = 39810.72 nM T39195 CSW48V 155557718 IC50 = 31.62 nM T39195 CNZ1K5 155559920 Ki > 10000 nM T39195 C6N0LM 155564043 Ki = 150 nM T39195 CM8XB1 155565537 IC50 = 794.33 nM T39195 D00LOL 970375 IC50 = 1290 nM T42025 D08QMX 5757 IC50 = 3.2 nM T42025 D0L4FS 5280961 IC50 = 395 nM T42025 CQ0IC4 63062 IC50 = 886 nM T42025 CJLH38 11154982 IC50 = 10 nM T42025 C4WO6B 11223355 IC50 = 210 nM T42025 C30IWO 11373378 IC50 = 750 nM T42025 C9BC0L 16732000 Ki > 10000 nM T42025 CN9L7G 46916268 EC50 = 1600 nM T42025 C5ZX4B 54597874 IC50 > 10000 nM T42025 CB54WI 71605373 IC50 = 436.4 nM T42025 CV9N4F 71605540 IC50 = 331.1 nM T42025 C56KSX 71605541 IC50 = 185 nM T42025 CYW9V0 71605542 IC50 = 150.6 nM T42025 CM07WE 71605543 IC50 = 19.1 nM T42025 C7EIS1 71605704 IC50 = 565.9 nM T42025 C7NBI8 71605705 IC50 = 120.7 nM T42025 C3LD2H 71605706 IC50 = 111.9 nM T42025 C3J5UW 71605707 IC50 = 41.2 nM T42025 C2URL4 134134246 IC50 > 10000 nM T42025 CD7NA5 134138492 IC50 > 10000 nM T42025 CP04WC 134144077 IC50 > 10000 nM T42025 CYG76M 134150509 IC50 > 10000 nM T42025 C89SMK 134152807 IC50 = 6950 nM T42025 C1O0IW 134153257 IC50 > 10000 nM T42025 C0Z4OD 134155524 IC50 > 10000 nM T42025 C58OUX 134155994 IC50 = 722 nM T42025 C3AF1G 135356810 IC50 = 350 nM T42025 CG6J2U 135356971 IC50 = 50 nM T42025 CM98IN 135356983 IC50 = 2250 nM T42025 CI2OM9 135399711 IC50 = 504 nM T42025 CH2K3S 135424843 IC50 = 1130 nM T42025 C67LAW 135427962 IC50 = 1017 nM T42025 C30QWY 135430315 IC50 = 455 nM T42025 CB3XM0 135438509 IC50 = 820 nM T42025 CVBN04 135446024 IC50 = 5235 nM T42025 CB5P0O 135461031 IC50 = 2345 nM T42025 CYJ96L 135508068 IC50 = 549 nM T42025 CA3F6J 135508229 IC50 = 98 nM T42025 CNXJ86 137628681 IC50 > 10000 nM T42025 CC6QT1 137632572 IC50 = 600 nM T42025 CA6J9P 137634677 IC50 = 550 nM T42025 CXJ8G2 137636516 IC50 = 1100 nM T42025 C6O5LB 137648454 IC50 = 300 nM T42025 C5ME8W 145964103 EC50 = 45 nM T42025 CA41IJ 145964137 EC50 = 2700 nM T42025 C0N3VX 145972148 EC50 = 31 nM T42025 CKTL80 145975927 EC50 = 20 nM T42025 C3P9HV 145977071 EC50 = 90 nM T42025 C0XYI1 145978085 EC50 = 630 nM T42025 C7VS5G 155511937 IC50 = 1330 nM T42025 CVCK17 155513135 IC50 = 861 nM T42025 C2PU1J 155513315 IC50 = 1980 nM T42025 CMQC26 155515404 IC50 = 2002 nM T42025 CP1L3J 155516697 IC50 = 2097 nM T42025 CSLJ15 155528850 IC50 = 2800 nM T42025 CC5HJ6 155535796 IC50 = 1017 nM T42025 CB3CY8 155538987 IC50 = 4540 nM T42025 CA5G2T 155551013 IC50 = 990 nM T42025 C7AJZ5 155559268 IC50 = 3040 nM T42025 C9KY5I 155562382 IC50 = 980 nM T42025 CWK95R 155565459 IC50 = 1045 nM T42025 CY71WP 155565677 IC50 = 1440 nM T42025 CMX67L 155567147 IC50 = 1648 nM T42025 D00QDE 135520118 IC50 = 56 nM T42025 D01TUB 135519319 IC50 = 213 nM T42025 D03CBX 135454802 IC50 = 212 nM T42025 D07XJC 135466462 IC50 = 641 nM T42025 D08SJL 135524856 IC50 = 1500 nM T42025 D09FWS 135430317 IC50 = 634 nM T42025 D09NFD 6852176 IC50 = 3500 nM T42025 D0I1AF 135438472 IC50 = 526 nM T42025 D0K7HR 135409729 IC50 = 504 nM T42025 D0RD6G 135453199 IC50 = 624 nM T42025 D0W1YT 135466468 IC50 = 88 nM T48940 D02PMO 60700 EC50 = 71.3 nM T48940 D07DJQ 10219 IC50 = 83 nM T48940 D07VLY 31703 EC50 = 120 nM T48940 D0M2QH 441852 EC50 = 20 nM T48940 D07AOL 16741 IC50 = 7500 nM T48940 D0AY8W 101913833 IC50 = 21 nM T48940 D0K0PG 16124726 IC50 = 2600 nM T48940 D0LK6V 54575622 IC50 = 280 nM T48940 C65JLT 3330 IC50 = 310 nM T48940 CMLZ97 6185 EC50 = 2000 nM T48940 C4Q7KS 92765 IC50 = 8.7 nM T48940 C7KJ3B 114917 IC50 = 8510 nM T48940 C37TUW 122838 IC50 = 12300 nM T48940 CSA18K 149138 IC50 > 20000 nM T48940 C5X1YU 160254 IC50 = 1360 nM T48940 C4IRY2 164676 IC50 = 6180 nM T48940 CYWS98 185848 IC50 > 30000 nM T48940 CJS21N 309568 IC50 > 30000 nM T48940 CMC10D 324099 IC50 = 3000 nM T48940 CS8B4Y 445420 IC50 = 6700 nM T48940 CJR6O1 562801 IC50 > 30000 nM T48940 C0JLU2 589919 IC50 = 560 nM T48940 CEN1R3 727149 IC50 > 30000 nM T48940 C62UTE 762138 IC50 = 5400 nM T48940 C32QWR 910367 IC50 > 30000 nM T48940 CJ5D7A 1278684 IC50 > 30000 nM T48940 CV9RT4 1278687 IC50 > 30000 nM T48940 CDM4E8 1363752 IC50 = 29000 nM T48940 CJ0R3B 2211000 IC50 = 280 nM T48940 C5O0PV 3494993 IC50 = 2500 nM T48940 CTM9S1 3801858 IC50 = 13900 nM T48940 CL0CT4 3906683 IC50 = 9900 nM T48940 CN59EU 3967295 IC50 > 30000 nM T48940 CFH6R1 4216314 IC50 = 10500 nM T48940 CCG53N 4567648 IC50 > 30000 nM T48940 C6TV3P 4770495 IC50 = 19100 nM T48940 CS7ED1 4770795 IC50 > 100000 nM T48940 CRL3T4 4771004 IC50 = 8100 nM T48940 C2OCJ7 4771616 IC50 = 8700 nM T48940 CF70TK 5124065 IC50 = 5000 nM T48940 CJFM37 5281419 IC50 = 3710 nM T48940 CJM8V5 5468522 IC50 = 6100 nM T48940 CJZ4E8 5489487 IC50 = 2200 nM T48940 C54WYM 5748528 IC50 = 9560 nM T48940 CYT08D 5748555 IC50 = 3230 nM T48940 CG23SW 9971020 IC50 = 3180 nM T48940 CE8KL2 9972857 IC50 > 30000 nM T48940 C8PRK4 10030510 IC50 = 320 nM T48940 CEY6O0 10039317 IC50 = 340 nM T48940 C28XBM 10055535 IC50 = 30 nM T48940 CP4M9D 10089207 IC50 > 30000 nM T48940 C43JMR 10250175 IC50 = 7200 nM T48940 C72MEI 10364986 IC50 = 200 nM T48940 CWUQ45 10439828 IC50 = 3 nM T48940 C0RU2G 10457340 IC50 = 200 nM T48940 CD25TE 11174259 EC50 = 400 nM T48940 CW5LU7 11325812 IC50 = 10000 nM T48940 C1JAC5 11425923 IC50 = 2290 nM T48940 CG8V9X 11429041 IC50 = 20000 nM T48940 C2JG9M 11843703 IC50 = 48.1 nM T48940 CQ90HV 12302705 IC50 = 1100 nM T48940 CZK16N 14539883 IC50 > 30000 nM T48940 CB42PF 14610613 IC50 = 7340 nM T48940 CK68ZD 14610678 IC50 = 8700 nM T48940 CJ3B2F 15378863 IC50 > 30000 nM T48940 CNI19E 15479637 IC50 = 8750 nM T48940 C7QJO4 15479638 IC50 = 8260 nM T48940 C3CKM1 15484930 IC50 = 10600 nM T48940 C72FQR 15605807 IC50 = 910 nM T48940 CIH7R0 15818782 IC50 > 50000 nM T48940 CSVZ40 16097752 IC50 = 593 nM T48940 CBT15H 16099424 IC50 = 20000 nM T48940 CN4C2I 16099425 IC50 = 20000 nM T48940 C9CIY2 16099426 IC50 > 30000 nM T48940 CF5YT3 16099427 IC50 > 30000 nM T48940 C76MRV 16099429 IC50 = 25000 nM T48940 C92MPD 16099430 IC50 = 30000 nM T48940 C2UV3B 16099431 IC50 = 15000 nM T48940 C97LRM 16099432 IC50 > 30000 nM T48940 CI0S6N 16124722 IC50 = 14080 nM T48940 C0YKL1 16124723 IC50 > 30000 nM T48940 CDO19C 16124724 IC50 = 23200 nM T48940 C0SG2C 16124727 IC50 = 400 nM T48940 C7J6QC 16124788 IC50 > 30000 nM T48940 CUL90W 16124789 IC50 > 30000 nM T48940 CYO1C5 16124850 IC50 = 4300 nM T48940 C3Y1TC 16124851 IC50 > 30000 nM T48940 CBT52L 16124923 IC50 > 30000 nM T48940 C4KLZ1 16124924 IC50 > 30000 nM T48940 CC01MW 16124925 IC50 > 30000 nM T48940 C5I6TJ 16124990 IC50 = 8200 nM T48940 CWX2K4 16124991 IC50 > 30000 nM T48940 C4D6LX 16124992 IC50 > 30000 nM T48940 C71CSU 16124996 IC50 > 30000 nM T48940 C5V7KM 16125063 IC50 = 12600 nM T48940 CJ3BG7 16125696 IC50 > 30000 nM T48940 C5I1YJ 19412490 IC50 = 81800 nM T48940 CU05IT 19412507 IC50 = 72000 nM T48940 C9O5FA 19467838 IC50 = 19400 nM T48940 CY9K6W 20055295 EC50 = 40 nM T48940 CI3QD6 20056162 IC50 > 30000 nM T48940 COV4Q3 21637526 IC50 = 2900 nM T48940 CQU5I0 21637535 IC50 = 500 nM T48940 C9LIB6 21773185 IC50 = 20000 nM T48940 C0V1KI 21773186 IC50 > 30000 nM T48940 C6I9YJ 21775613 IC50 = 20000 nM T48940 C0S6VL 23424966 IC50 = 200 nM T48940 C5JC7D 23427322 IC50 > 30000 nM T48940 CLES79 23642918 IC50 = 7300 nM T48940 C59KHO 24179737 IC50 = 5100 nM T48940 CSFN10 24853811 IC50 = 29000 nM T48940 C8VS9Y 24882418 IC50 > 50000 nM T48940 CX2P1E 25158444 IC50 = 2600 nM T48940 CU4ZH9 25169523 IC50 = 3000 nM T48940 C3R1OG 25208124 IC50 > 30000 nM T48940 CF15DX 25208125 IC50 > 30000 nM T48940 C5HL9G 35534418 IC50 > 100000 nM T48940 CL60AQ 44139361 EC50 = 600 nM T48940 CRXW65 44229629 IC50 = 26300 nM T48940 C2YOZ1 44420796 IC50 > 30000 nM T48940 CD7AB1 44425164 IC50 > 20000 nM T48940 C2M4YU 44425165 IC50 = 12700 nM T48940 C8W1NF 44425166 IC50 > 20000 nM T48940 C9TK1Z 44445342 IC50 = 4500 nM T48940 CR5I0B 44445343 IC50 = 2400 nM T48940 C4Z7JA 44445792 IC50 = 3900 nM T48940 C1LCQ2 44450293 IC50 = 5700 nM T48940 CZNL75 44450330 IC50 > 50000 nM T48940 CQP80T 44457182 EC50 = 13000 nM T48940 CY1O5V 44457186 EC50 = 8000 nM T48940 C4R7SH 44457187 EC50 = 6000 nM T48940 C0HYD9 44575507 IC50 = 13 nM T48940 CK0VC9 44604734 IC50 = 10000 nM T48940 C3E5FX 44604735 IC50 = 7800 nM T48940 CAX5R1 44604736 IC50 = 8600 nM T48940 CY6MG5 44604940 IC50 = 10000 nM T48940 C36MXH 44604945 IC50 = 10000 nM T48940 CHAZ63 44605144 IC50 = 20000 nM T48940 C1R9TY 44605146 IC50 = 20000 nM T48940 CG41IA 44605147 IC50 = 20000 nM T48940 CE4L7N 44605148 IC50 = 20000 nM T48940 CDV57K 44605150 IC50 = 20000 nM T48940 C45RQB 45485201 IC50 = 8550 nM T48940 CG4MJ0 46208134 IC50 = 380 nM T48940 C5IXA7 46208135 IC50 = 350 nM T48940 C4OQ8B 46208266 IC50 = 1440 nM T48940 C7D8OC 46881366 IC50 = 7700 nM T48940 CG6I2T 46888567 IC50 = 12 nM T48940 CRHA93 50908588 IC50 = 2000 nM T48940 CW6FT9 51040687 IC50 = 2230 nM T48940 C4E8UG 51040688 IC50 = 1720 nM T48940 C8NPQ2 51040689 IC50 = 4120 nM T48940 CLDH27 51040903 IC50 = 5110 nM T48940 C58FMU 51040904 IC50 = 830 nM T48940 C46OWL 51040905 IC50 = 2060 nM T48940 C69CHX 51040906 IC50 = 18400 nM T48940 CS2L0N 51040907 IC50 = 15700 nM T48940 CY3IQ6 51041102 IC50 = 6310 nM T48940 CY39VN 51041103 IC50 = 7420 nM T48940 CN60AL 53318796 IC50 = 2710 nM T48940 C0QCU6 53320112 IC50 = 3250 nM T48940 C7LUZ9 53321420 IC50 = 4630 nM T48940 CXM45T 53322741 IC50 = 6760 nM T48940 CRY0O7 53324072 IC50 = 3400 nM T48940 CNJ59Y 53325382 IC50 = 5310 nM T48940 CX5A2S 53326644 IC50 = 8210 nM T48940 C4VO7M 53467839 IC50 = 0.47 nM T48940 CNUE41 53472867 IC50 = 500 nM T48940 C3C1PM 53483997 IC50 = 508 nM T48940 CR1B9H 53483998 IC50 = 656 nM T48940 CE40RG 53483999 IC50 = 532 nM T48940 CE4FC0 54575618 IC50 = 500 nM T48940 CLY0Z3 54575619 IC50 = 600 nM T48940 C73YAJ 54575620 IC50 = 306 nM T48940 CDN1I8 54575621 IC50 = 600 nM T48940 C7Q1PX 54575623 IC50 = 478 nM T48940 C7EF6H 54575686 IC50 = 378 nM T48940 CZU9S8 56662022 IC50 = 2100 nM T48940 CKA6B8 56662203 IC50 = 1097 nM T48940 CVTJ72 56662204 IC50 = 1011 nM T48940 CI8A9V 56669104 IC50 > 25000 nM T48940 CU3Q5V 56675807 IC50 = 3000 nM T48940 CGNZ39 56675943 IC50 = 4000 nM T48940 C5HU8O 56679124 IC50 = 1500 nM T48940 CNAH02 56679260 IC50 = 731 nM T48940 C85IEA 56679261 IC50 = 672 nM T48940 C4D5FP 56682420 IC50 = 16800 nM T48940 CZK23O 56682564 IC50 = 4200 nM T48940 CT72DG 56925644 IC50 = 2200 nM T48940 CVC71E 56925645 IC50 = 2200 nM T48940 CONB80 56925651 IC50 = 3000 nM T48940 CHCM59 56925766 IC50 = 8500 nM T48940 CJ7IU1 56925767 IC50 > 25000 nM T48940 CXD81G 56925768 IC50 > 25000 nM T48940 CV65WF 56925769 IC50 > 25000 nM T48940 CU89KS 56925770 IC50 > 25000 nM T48940 CIB79E 56925886 IC50 = 5000 nM T48940 C9YN0C 56925887 IC50 = 8400 nM T48940 CQ95IY 56925888 IC50 = 2600 nM T48940 CHA9F1 56925889 IC50 = 1300 nM T48940 CTL17N 56925890 IC50 = 3300 nM T48940 CJ75MH 56925891 IC50 = 3500 nM T48940 CUZ72W 56925992 IC50 = 3400 nM T48940 C29IUA 56925993 IC50 = 1500 nM T48940 C1YVP9 56926089 IC50 = 9100 nM T48940 CB62JK 56926090 IC50 = 1500 nM T48940 CA9HW0 56926091 IC50 = 8200 nM T48940 C81KXF 56926093 IC50 = 2500 nM T48940 CG3WJ4 56926179 IC50 > 25000 nM T48940 C4GIL9 56926181 IC50 = 1300 nM T48940 CZ2T1Y 56926182 IC50 = 900 nM T48940 C9B8OJ 56926183 IC50 > 25000 nM T48940 CS9B4Q 56926184 IC50 = 800 nM T48940 CZ0SI5 56926270 IC50 = 6200 nM T48940 CP7TV8 56926271 IC50 = 6600 nM T48940 CZW1B3 56926272 IC50 = 700 nM T48940 C5B6IH 56926273 IC50 = 5700 nM T48940 CM86YP 56926274 IC50 = 400 nM T48940 CDMH43 56926275 IC50 = 13400 nM T48940 C3QS7C 56926368 IC50 > 25000 nM T48940 C8P5YI 56926369 IC50 = 5000 nM T48940 C3W6NL 56926370 IC50 = 6400 nM T48940 C5LVS7 56926371 IC50 = 900 nM T48940 C3NFH8 56926372 IC50 = 3400 nM T48940 CT45QP 56926373 IC50 = 6500 nM T48940 CBR2Q1 56926475 IC50 = 900 nM T48940 C8X2VW 56926476 IC50 = 900 nM T48940 C4FH2O 56926479 IC50 = 1400 nM T48940 C9POA3 56926480 IC50 = 1800 nM T48940 CQ2X3G 56926595 IC50 = 5800 nM T48940 CU4D7I 56926596 IC50 = 1100 nM T48940 CD1F4S 57392062 IC50 = 63 nM T48940 CLYW05 57394694 IC50 = 1600 nM T48940 C7A6HY 57395543 IC50 = 68 nM T48940 C6OMU3 70684272 IC50 = 8000 nM T48940 C76XIO 70685494 IC50 = 11 nM T48940 CBR0A3 70686427 IC50 = 4800 nM T48940 C42ISF 70686428 IC50 = 2700 nM T48940 CI3F6L 70688533 IC50 = 2200 nM T48940 CU15GB 70694769 IC50 = 6600 nM T48940 CA9SC1 70694770 IC50 = 4800 nM T48940 CF56SV 70694771 IC50 = 7200 nM T48940 CF97GN 70696811 IC50 = 3200 nM T48940 C9UB6K 70696815 IC50 = 3800 nM T48940 C93OKA 71453127 IC50 = 2300 nM T48940 C8BU6Z 71454859 IC50 = 1200 nM T48940 CQ6DX9 71456630 IC50 = 4200 nM T48940 CF9WJ8 71620853 IC50 = 7.9 nM T48940 C2R1QU 73349944 IC50 = 5940 nM T48940 CP79XF 91668262 IC50 = 690 nM T48940 CD83HY 92672401 IC50 > 10000 nM T48940 C3L7DC 117855105 IC50 = 430 nM T48940 CDT9A3 118714262 IC50 = 2200 nM T48940 C53XSK 118714263 IC50 > 20000 nM T48940 CL2D1Q 118714264 IC50 = 4000 nM T48940 CVB89I 118714429 IC50 > 10000 nM T48940 C27HZP 118714430 IC50 = 230 nM T48940 CCD5I8 118714431 IC50 = 4500 nM T48940 CFPU93 118714432 IC50 = 1600 nM T48940 C0I9SU 118714433 IC50 = 880 nM T48940 CYRH54 118714434 IC50 = 2500 nM T48940 CW6SN7 118714435 IC50 = 2200 nM T48940 CIT5S8 118714437 IC50 = 13 nM T48940 CEI47B 118714438 IC50 = 7.9 nM T48940 C4Q3RC 118714439 IC50 = 110 nM T48940 C0FMS7 118714440 IC50 = 14 nM T48940 CQH62A 118714441 IC50 = 120 nM T48940 C6RV9T 118714442 IC50 = 3.3 nM T48940 C1TYS7 118714443 IC50 = 13 nM T48940 CANH91 118714444 IC50 = 30 nM T48940 CH2BK8 118714445 IC50 = 35 nM T48940 CBD97Q 118714446 IC50 = 34 nM T48940 C5HOW1 118714447 IC50 = 3.1 nM T48940 C19CQT 118714448 IC50 > 200 nM T48940 CFVM09 118714449 IC50 = 0.97 nM T48940 CN5R3M 118714450 IC50 = 5.8 nM T48940 C1FMC2 118714451 IC50 = 2.6 nM T48940 C4XP3T 118714452 IC50 = 1.1 nM T48940 CKQT34 118729528 IC50 > 100000 nM T48940 CIL4V1 118729529 IC50 > 100000 nM T48940 C0EFK5 118729530 IC50 = 71600 nM T48940 CCZ45B 118729531 IC50 > 100000 nM T48940 CI0GF8 122192794 IC50 = 2110 nM T48940 C5H2MX 122192795 IC50 > 10000000 nM T48940 CNF4Z9 122192796 IC50 = 3700 nM T48940 CT3I1N 122192797 IC50 = 1930 nM T48940 CWFP59 122192798 IC50 = 590 nM T48940 CDVF09 134132602 IC50 = 9400 nM T48940 CY28SJ 134133716 IC50 = 6500 nM T48940 CFR62T 134136549 IC50 = 56000 nM T48940 CRW5O0 134139477 IC50 = 61000 nM T48940 C93CEI 134139559 IC50 = 17000 nM T48940 CH75UQ 134140118 IC50 = 7400 nM T48940 CU62OY 134142080 IC50 = 3700 nM T48940 C7NTX6 134143336 IC50 = 25000 nM T48940 CZR2P0 134145784 IC50 = 75000 nM T48940 CLG97I 134147044 IC50 = 39000 nM T48940 CRN4Z0 134149171 IC50 = 9100 nM T48940 CKH87B 134155395 IC50 = 70000 nM T48940 CC8WR6 135400930 IC50 = 3400 nM T48940 C2N4WE 135830852 IC50 = 2900 nM T48940 C7SQC6 135846960 IC50 = 1700 nM T48940 CMJ23G 136075559 IC50 > 30000 nM T48940 CYF1R9 136193084 IC50 = 2700 nM T48940 CV39WX 136268869 IC50 = 14500000 nM T48940 CGFU84 136268871 IC50 = 15900 nM T48940 CN5SJ1 136268872 IC50 = 18900000 nM T48940 CPY3M7 136268873 IC50 = 10100 nM T48940 C49QMW 136268879 IC50 = 23900 nM T48940 CM4O5B 136268880 IC50 = 3800000 nM T48940 CK96MF 137036807 IC50 > 30000 nM T48940 CCFS85 137036808 IC50 > 30000 nM T48940 C1BME9 137036809 IC50 > 30000 nM T48940 C75PZK 137036810 IC50 > 30000 nM T48940 C5J3RC 137036811 IC50 > 30000 nM T48940 C85EID 137036812 IC50 > 30000 nM T48940 C07MVZ 137036813 IC50 > 30000 nM T48940 C8XLD3 137036814 IC50 > 30000 nM T48940 C8MNO6 137036815 IC50 > 30000 nM T48940 CJK2M1 137036816 IC50 > 30000 nM T48940 C9USP2 137036817 IC50 > 30000 nM T48940 D00REK 5712 IC50 = 48400 nM T48940 D01NUT 5467256 IC50 = 8760 nM T48940 D01OQW 9959532 IC50 > 30000 nM T48940 D06ZWX 6197 IC50 = 36 nM T48940 D08VRV 45485203 IC50 = 9540 nM T48940 D09WED 45485202 IC50 = 6420 nM T48940 D0E1ZS 5281297 IC50 = 6270 nM T48940 D0H1WV 45273151 IC50 = 6070 nM T39054 CG80HD 6457 Ki > 1000000 nM T39054 CD85ZQ 65159 Ki > 1000000 nM T39054 C9V7XZ 69925 Ki > 1000000 nM T39054 CM70AT 252390 Ki = 1000000 nM T39054 C0BUG1 300719 Ki > 1000000 nM T39054 C5WR6U 4369390 Ki = 457000 nM T39054 C7X5HM 9872431 Ki = 300 nM T39054 CU6H2R 10405129 Ki = 119000 nM T39054 C9AB7C 10406444 Ki > 1000000 nM T39054 C7HZ4R 11036334 Ki > 1000000 nM T39054 C35GBD 11091653 Ki = 157000 nM T39054 CE83KQ 11431328 Ki = 46000 nM T39054 CRC0T4 11487560 Ki > 1000000 nM T39054 CZ83RF 11495602 Ki > 1000000 nM T39054 CW43EV 11503449 Ki = 21000 nM T39054 CK2D9P 11508549 Ki > 1000000 nM T39054 C8B1CO 11518135 Ki = 476000 nM T39054 C3XVF1 11521261 Ki > 1000000 nM T39054 CZO0K7 11525876 Ki > 1000000 nM T39054 CQBZ68 11536503 Ki > 1000000 nM T39054 CMSV60 11568040 Ki > 1000000 nM T39054 CFW21T 11568685 Ki > 1000000 nM T39054 CX34SJ 11596749 Ki = 313000 nM T39054 C1ZT2L 11597370 Ki > 1000000 nM T39054 CO75DF 11597721 Ki = 260000 nM T39054 C2UHA3 11600743 Ki > 1000000 nM T39054 CQOL87 11601721 Ki = 311000 nM T39054 CX1A7W 11602125 Ki > 1000000 nM T39054 CQ90LJ 11604271 Ki > 1000000 nM T39054 CJ4T2F 11611914 Ki > 1000000 nM T39054 CS87TE 11612392 Ki > 1000000 nM T39054 CX7V6G 11612667 Ki > 1000000 nM T39054 CDN05O 11626095 Ki = 25000 nM T39054 CL7P5R 11627408 Ki = 74000 nM T39054 CS46FV 11633797 Ki > 1000000 nM T39054 CI67CB 11637769 Ki = 73000 nM T39054 C4XKI1 11640066 Ki > 1000000 nM T39054 CT48RO 11645202 Ki > 1000000 nM T39054 CZ9Q5W 11650008 Ki > 1000000 nM T39054 C1EK7Y 11655779 Ki = 383000 nM T39054 C3B8ON 11659618 Ki > 1000000 nM T39054 CQ17DI 11662581 Ki = 135000 nM T39054 C9L1YB 11678639 Ki > 1000000 nM T39054 C6X8LG 11680992 Ki = 63000 nM T39054 CUMO12 11684941 Ki > 1000000 nM T39054 CYCJ41 11695395 Ki > 1000000 nM T39054 CJ41GW 11697478 Ki = 324000 nM T39054 C4J5OG 11701790 Ki = 898000 nM T39054 C9FY5C 11719489 Ki > 1000000 nM T39054 CZ7X6J 12353387 Ki > 1000000 nM T39054 C0XIS9 13711960 Ki = 18000 nM T39054 CC5YM2 14260322 Ki > 1000000 nM T39054 C7IF2B 14308789 Ki = 56400 nM T39054 CQ69MX 14426909 Ki = 157000 nM T39054 CJ2LH3 14680571 Ki > 1000000 nM T39054 CL19NZ 14680572 Ki > 1000000 nM T39054 C93XDA 15277759 Ki = 806000 nM T39054 C38TCQ 18368821 Ki = 1000000 nM T39054 CTE98V 25266093 Ki > 1000000 nM T39054 C4P2QK 25266094 Ki > 1000000 nM T39054 C7ZXT1 25266095 Ki > 1000000 nM T39054 C2X4FV 25266098 Ki > 1000000 nM T39054 CRAC39 25266432 Ki > 1000000 nM T39054 C6BV8F 25266433 Ki > 1000000 nM T39054 C32YKJ 25266436 Ki > 1000000 nM T39054 C57VDQ 25266437 Ki > 1000000 nM T39054 C04KDB 42624707 Ki > 1000000 nM T39054 CG80LO 44403852 Ki = 46000 nM T39054 C15WGH 44403871 Ki > 1000000 nM T39054 C12SWP 44403872 Ki = 808000 nM T39054 C5B6LE 44403876 Ki > 1000000 nM T39054 C24UGC 44403880 Ki > 1000000 nM T39054 C8WI9O 44403881 Ki = 232000 nM T39054 C38EQZ 44403896 Ki > 1000000 nM T39054 CWF18U 44403897 Ki > 1000000 nM T39054 CZS36L 44403901 Ki > 1000000 nM T39054 CB2K5Q 44403902 Ki > 1000000 nM T39054 CF5X0D 44403907 Ki > 1000000 nM T39054 COB5S9 44403909 Ki = 469000 nM T39054 CU05XL 44403910 Ki > 1000000 nM T39054 CNO6X1 44403912 Ki > 1000000 nM T39054 C8M1RT 44403913 Ki > 1000000 nM T39054 C5CH8F 44403924 Ki = 457000 nM T39054 C57YCL 44403929 Ki > 1000000 nM T39054 C9NO6D 44403930 Ki > 1000000 nM T39054 C8LT1P 44403931 Ki = 799000 nM T39054 CSY15V 44403932 Ki = 350000 nM T39054 C6SQI9 44403933 Ki = 298000 nM T39054 C28NCK 44403934 Ki > 1000000 nM T39054 CL03MN 44403935 Ki > 1000000 nM T39054 CVF0J8 44413521 Ki = 909000 nM T39054 C26KJE 44413566 Ki = 636000 nM T39054 CYG75F 44413618 Ki = 496000 nM T39054 CJ3C4Q 44544449 IC50 = 21 nM T39054 C6AO9H 44544550 IC50 = 40 nM T39054 CCRX17 44582171 Ki > 1000000 nM T39054 CX1M5F 44622388 IC50 = 1300 nM T39054 C4BGR0 44622389 IC50 = 2500 nM T39054 CX6RS4 45107976 IC50 = 290 nM T39054 C6UOD2 45108053 IC50 = 600 nM T39054 C5MZC4 45108054 IC50 > 1000 nM T39054 C3XTQ9 45108084 IC50 > 1000 nM T39054 CIYO05 45108085 IC50 = 350 nM T39054 C4S5WT 45108086 IC50 > 1000 nM T39054 CC9Z3U 45108087 IC50 = 10000 nM T39054 C27KHT 49786956 IC50 = 320 nM T39054 CNWM80 49795041 EC50 = 5100 nM T39054 CTI4K0 53233170 IC50 = 62 nM T39054 C9X4RS 53248784 Ki > 100000 nM T39054 CO6A8Q 53248785 Ki > 100000 nM T39054 CST5D7 53248786 Ki > 100000 nM T39054 C19WZD 54580005 Ki > 100000 nM T39054 C47MQI 54581004 Ki > 100000 nM T39054 C1RCN5 54581005 Ki > 100000 nM T39054 C12BFA 54582039 Ki > 100000 nM T39054 CM2X3I 54582040 Ki > 100000 nM T39054 CM0JS9 54582986 Ki > 100000 nM T39054 C7HK6P 54582987 Ki > 100000 nM T39054 CX4N9T 54583982 Ki > 100000 nM T39054 C8IVG9 54583983 Ki > 100000 nM T39054 CASG08 54583984 Ki = 90000 nM T39054 CEI0P7 54584925 Ki > 100000 nM T39054 CU26MC 54584926 Ki = 98000 nM T39054 CXUF05 54585889 Ki > 100000 nM T39054 C5JQ9P 54585890 Ki > 100000 nM T39054 CGQA63 54586862 Ki > 100000 nM T39054 C37ZCX 54586863 Ki > 100000 nM T39054 C1ZSJ3 54753440 Ki > 100000 nM T39054 CYT87V 54753630 Ki = 49000 nM T39054 CJ35MZ 57385001 IC50 = 97000 nM T39054 C7B4CP 57385248 IC50 > 30000 nM T39054 CH0JI4 57385249 IC50 = 22000 nM T39054 CM3X9G 57385250 IC50 > 30000 nM T39054 C8RNI3 57385251 IC50 > 30000 nM T39054 CS45NE 57385252 IC50 > 30000 nM T39054 CR7B9E 57385253 IC50 > 30000 nM T39054 CW02SJ 57385254 IC50 > 30000 nM T39054 CSG56M 57385497 IC50 > 30000 nM T39054 C2FXH8 57385498 IC50 = 7300 nM T39054 C4IA9M 57385499 IC50 > 30000 nM T39054 CCE5B4 57385500 IC50 = 30000 nM T39054 CU5SV9 57385501 IC50 > 30000 nM T39054 C46VEN 57385502 IC50 > 30000 nM T39054 CON98H 57385503 IC50 > 30000 nM T39054 CJC04P 57385504 IC50 > 30000 nM T39054 C9LB8O 57385739 IC50 > 30000 nM T39054 C48UNT 57385740 IC50 = 16000 nM T39054 C7FA0W 57385741 IC50 > 30000 nM T39054 C4MN0X 57385742 IC50 = 21000 nM T39054 C6U5OD 57385743 IC50 > 30000 nM T39054 CL68QM 57385744 IC50 = 1100 nM T39054 CX1NZ3 57385745 IC50 = 580 nM T39054 C8DR1A 57386012 IC50 > 1000 nM T39054 CT12AB 57386014 IC50 = 150 nM T39054 CGN54B 57386015 IC50 > 1000 nM T39054 CYHC93 57386270 IC50 = 9400 nM T39054 CAM4H3 57386271 IC50 = 280 nM T39054 CS0H9Z 57386272 IC50 = 310 nM T39054 CA38OZ 57386525 IC50 > 1000 nM T39054 CK9A7F 57386526 IC50 > 1000 nM T39054 CYLU51 57386527 IC50 = 19500 nM T39054 CAF81E 57386528 IC50 = 1200 nM T39054 CM47HD 57386529 IC50 = 18200 nM T39054 CAE62M 57386786 IC50 = 9400 nM T39054 CSH81D 57386787 IC50 = 4500 nM T39054 CZ8T6U 57386788 IC50 = 5700 nM T39054 CV1FH8 57386789 IC50 = 35 nM T39054 CWK97J 57387036 IC50 = 340 nM T39054 CP3XL5 57387037 IC50 = 2500 nM T39054 CSIC05 60154749 EC50 = 140 nM T39054 CT3F6L 60154750 EC50 = 120 nM T39054 CQX5W8 60154751 IC50 = 73 nM T39054 CF8XO1 60154753 IC50 = 340 nM T39054 CFA31N 60154848 IC50 = 28 nM T39054 CY8F4G 60154849 EC50 = 200 nM T39054 C1M5AW 60154850 EC50 = 49 nM T39054 CP5M3A 60154851 EC50 = 930 nM T39054 CGXH67 60154852 EC50 = 610 nM T39054 CP2OU4 60154853 IC50 = 410 nM T39054 CX1SH3 60154936 IC50 = 39 nM T39054 CA53KC 60154937 EC50 = 150 nM T39054 C8R3CK 60154938 IC50 = 82 nM T39054 CY5Q3N 60156015 EC50 = 2600 nM T39054 C2IS7J 60156016 EC50 = 2600 nM T39054 CUN50O 60156119 EC50 = 3130 nM T39054 CA9ZX6 60195478 EC50 = 1100 nM T39054 CA10IJ 60195479 IC50 = 740 nM T39054 C7GZV4 60195559 IC50 > 10000 nM T39054 CL39TW 60195560 IC50 = 1600 nM T39054 C1UZS7 60195561 IC50 > 10000 nM T39054 C1Y4PV 60195562 IC50 = 3500 nM T39054 CLE14Y 60195563 IC50 = 5700 nM T39054 CS5PH3 60195564 IC50 = 4100 nM T39054 C4X1IU 60195565 IC50 > 10000 nM T39054 CFM8B6 60195639 IC50 = 390 nM T39054 CB1X4Q 60195640 IC50 = 210 nM T39054 CB1N6O 60195641 IC50 = 58 nM T39054 C57NBE 60195642 IC50 = 870 nM T39054 CDM85V 60195643 IC50 = 29 nM T39054 CG5H9Q 60195644 IC50 = 720 nM T39054 C8LGQ0 60195725 IC50 = 150 nM T39054 CQ54BT 60195726 IC50 > 1000 nM T39054 C5OC4S 60195727 IC50 = 170 nM T39054 C6HN9L 60195728 IC50 = 67 nM T39054 C83QGA 60195729 IC50 = 350 nM T39054 CNW78V 68699325 Ki > 1000000 nM T39054 CFYS45 70686348 IC50 = 3100 nM T39054 CC6BV1 70692586 IC50 = 230 nM T39054 C82WOZ 71449722 IC50 > 1000 nM T39054 C0K1XQ 71455073 IC50 = 210 nM T39054 CBO2F4 71456873 IC50 = 630 nM T39054 CG0FP7 71456874 IC50 > 1000 nM T39054 CD57XQ 71458726 IC50 = 150 nM T39054 CPT16Z 71460544 IC50 = 360 nM T39054 CW7RI9 71462256 IC50 = 550 nM T39054 CLK52V 72163617 Ki = 1000000 nM T39054 C4TPU0 72163618 Ki = 286000 nM T39054 CN3X2F 72163747 Ki = 1000000 nM T39054 C90MAV 72163748 Ki = 1000000 nM T39054 CV1PL9 72163749 Ki > 100000 nM T39054 C3BW1Y 73347672 Ki = 63000 nM T39054 CFR0P6 73350769 Ki = 10000 nM T39054 CB36MW 73353733 Ki = 1000000 nM T39054 C6CYK5 136254270 IC50 = 3300 nM T39054 D01SLZ 11704530 Ki = 5200 nM T39054 D0E2IH 11750725 Ki = 17000 nM T39054 D0K4DP 11683928 Ki = 5700 nM T39054 D0W5QR 11589642 Ki = 1400 nM T39054 D0Z9TM 448381 IC50 = 15000 nM T62431 D04AIT 5280445 EC50 = 4500 nM T62431 D04LVK 57379345 IC50 = 3050 nM T62431 D0AZ3C 5291 IC50 = 5000 nM T62431 D0K8KX 5280343 EC50 = 35000 nM T62431 D0OB0F 5328940 IC50 = 52 nM T62431 D0V8HJ 11671467 IC50 = 17 nM T62431 D02NNV 3038525 IC50 > 5000 nM T62431 D03HUX 49792852 IC50 > 10000 nM T62431 D03LWG 53235510 IC50 = 5358 nM T62431 D06DMQ 59472121 Ki = 190 nM T62431 D06KTJ 53252276 IC50 = 3.2 nM T62431 D07EHV 44814409 IC50 > 10000 nM T62431 D07HPJ 11476171 IC50 > 10000 nM T62431 D0E3TC 44259 IC50 < 0.1 nM T62431 D0G9AW 59473233 IC50 = 7.7 nM T62431 D0H2HZ 60194098 IC50 = 199.53 nM T62431 D0L4FS 5280961 IC50 = 39000 nM T62431 D0O0LS 25141092 IC50 > 1000 nM T62431 D0O6VZ 25254071 IC50 = 134 nM T62431 D0R9IU 44462758 IC50 = 1 nM T62431 D0S6TK 11213558 EC50 = 10 nM T62431 D0OE4F 4369496 Ki = 160 nM T62431 D08DBE 10344820 Ki = 1.8 nM T62431 D0T3ME 156422 IC50 > 20000 nM T62431 C8YI7Z 348911 IC50 = 5900000 nM T62431 CX0JA5 383690 IC50 = 14000 nM T62431 CNA8K3 718278 IC50 = 3800 nM T62431 CKND39 745199 EC50 = 5810 nM T62431 C7T1NS 802942 EC50 = 1430 nM T62431 COP6W0 1099108 EC50 = 1670 nM T62431 CHE8K4 1301845 IC50 > 200000 nM T62431 CR8QS9 1365090 IC50 = 4000 nM T62431 CSA3W9 1723820 IC50 = 3400 nM T62431 CY8FQ5 1776659 IC50 = 28400 nM T62431 CUZ6M1 2063494 IC50 = 8000000 nM T62431 CY35GB 2241431 IC50 = 57000 nM T62431 C25GNU 2877671 IC50 = 1900 nM T62431 CD02GY 4369033 IC50 = 20000 nM T62431 CUE64R 5329179 IC50 > 500000 nM T62431 CHA68G 5329180 IC50 > 500000 nM T62431 CNTD47 5329181 IC50 > 500000 nM T62431 CYFD81 5329182 IC50 > 500000 nM T62431 C21IKR 5329183 IC50 > 500000 nM T62431 C45ZME 5329185 IC50 > 500000 nM T62431 C5U7DB 5329186 IC50 > 500000 nM T62431 CQ6X8M 5329189 IC50 > 500000 nM T62431 C5HG9S 5329194 IC50 > 500000 nM T62431 CHV5Y6 5329195 IC50 > 500000 nM T62431 C3DOZ9 5329196 IC50 = 464000 nM T62431 CT61MB 5329197 IC50 > 500000 nM T62431 C6OT4G 5329198 IC50 > 500000 nM T62431 CROF47 5329199 IC50 > 500000 nM T62431 CHNM67 5329200 IC50 > 500000 nM T62431 C1G6ZU 5329201 IC50 > 500000 nM T62431 CA2HW9 5329202 IC50 > 500000 nM T62431 C30CUW 5329203 IC50 > 500000 nM T62431 C0UY4Q 5329204 IC50 > 500000 nM T62431 C3QIN5 5329205 IC50 > 500000 nM T62431 C5OBU1 5329206 IC50 > 500000 nM T62431 C2GKT3 5329207 IC50 = 452000 nM T62431 CKB23P 5329209 IC50 > 500000 nM T62431 CDL19N 5329212 IC50 = 302000 nM T62431 CI03PS 5329214 IC50 > 500000 nM T62431 C43NAT 5329215 IC50 > 500000 nM T62431 C9D3WP 5329216 IC50 > 500000 nM T62431 CS2I1H 5329217 IC50 > 500000 nM T62431 CQ70YG 5329218 IC50 > 500000 nM T62431 C6OL3X 5329220 IC50 > 500000 nM T62431 C2J4ZO 5329221 IC50 > 500000 nM T62431 CO87DJ 5329222 IC50 > 500000 nM T62431 C5LW1G 5329223 IC50 = 323000 nM T62431 CRB3S4 5329224 IC50 = 288000 nM T62431 CU68QR 5329225 IC50 = 250000 nM T62431 C4P7QH 5329226 IC50 = 318000 nM T62431 CWF7K8 5329227 IC50 > 500000 nM T62431 CJ6VE0 5329228 IC50 > 500000 nM T62431 C87VQB 5353854 IC50 = 14 nM T62431 C13KBC 5730111 IC50 = 120 nM T62431 C7WI1P 6326454 IC50 > 500000 nM T62431 CLB02J 6326455 IC50 > 500000 nM T62431 CZK47S 6326456 IC50 > 500000 nM T62431 CS23WK 6326457 IC50 > 500000 nM T62431 CR59JT 6326458 IC50 > 500000 nM T62431 CN1GO8 6326459 IC50 = 472000 nM T62431 CY4WT0 6326460 IC50 > 500000 nM T62431 CEW21T 6326461 IC50 = 397000 nM T62431 C3PNU9 6326462 IC50 > 500000 nM T62431 CLTQ35 6326463 IC50 = 433000 nM T62431 CU6S2L 6326464 IC50 > 500000 nM T62431 CNE5U9 8721605 IC50 = 27000 nM T62431 CI7JF8 9799509 IC50 = 10000 nM T62431 CTR6H5 9817349 IC50 = 30 nM T62431 CQVR76 9818573 IC50 = 34 nM T62431 C9VJG3 9820317 IC50 = 145 nM T62431 CLC0D4 9820420 IC50 = 8 nM T62431 CS1ET2 9836081 IC50 = 2000 nM T62431 CXQ9J0 9856983 Ki = 8 nM T62431 C9JC1G 9866765 IC50 = 2300 nM T62431 CM5Z8X 9869943 IC50 > 40000 nM T62431 C5DQF7 9902848 IC50 = 500 nM T62431 CT7O3P 9925060 IC50 = 500 nM T62431 C8SKR0 9952136 Ki = 10 nM T62431 CP9VK7 9965312 IC50 = 1000 nM T62431 CC2G8M 9968856 IC50 = 1000 nM T62431 CM15ZX 9968957 IC50 = 570 nM T62431 C3BL8S 9979898 IC50 = 9 nM T62431 C84LCW 9985193 IC50 > 500000 nM T62431 CO8CY4 10000020 IC50 = 5 nM T62431 CUY0F8 10005715 IC50 = 690 nM T62431 CGOT13 10022152 IC50 = 9 nM T62431 C4JO8F 10028975 IC50 = 28 nM T62431 C1O4GZ 10031003 IC50 > 500000 nM T62431 CGZC98 10044189 IC50 > 100000 nM T62431 C7YD1X 10048045 IC50 > 25000 nM T62431 CL9D6V 10084407 IC50 = 285000 nM T62431 CCW7U3 10097544 IC50 = 380 nM T62431 CO5G3R 10125483 IC50 = 420 nM T62431 C8YHF6 10125658 IC50 = 260 nM T62431 C8OE9N 10125723 IC50 = 90 nM T62431 C3K9ZV 10126020 IC50 = 890 nM T62431 CD1JN8 10149490 EC50 = 500 nM T62431 C7RUX6 10149633 IC50 = 140 nM T62431 CH3FD0 10149940 IC50 = 43 nM T62431 CLFN09 10150032 IC50 = 830 nM T62431 C1YE4U 10150080 IC50 = 210 nM T62431 CIO31T 10171604 IC50 = 230 nM T62431 C6VTK0 10172273 IC50 = 310 nM T62431 CGJ1A3 10193068 IC50 = 850 nM T62431 CVE31F 10193693 IC50 = 260 nM T62431 C5RZT2 10193837 IC50 = 900 nM T62431 CIQS71 10194027 IC50 = 330 nM T62431 CXOP81 10200390 Ki = 7.5 nM T62431 COY0K6 10214743 IC50 = 140 nM T62431 CWF1J9 10215022 EC50 = 460 nM T62431 C1X8OT 10215165 IC50 = 34 nM T62431 CMD8H6 10215299 IC50 = 72 nM T62431 C9S7HY 10236571 IC50 = 190 nM T62431 C4GHO6 10236578 IC50 = 500 nM T62431 C9JPR2 10236713 IC50 = 200 nM T62431 CSGD16 10246246 IC50 > 7000 nM T62431 C97GRN 10248747 IC50 > 100000 nM T62431 CDZ62G 10258706 IC50 = 38000 nM T62431 CBRA16 10286183 IC50 = 440 nM T62431 C79JMU 10286233 IC50 = 63 nM T62431 CU9O4G 10286428 IC50 = 1200 nM T62431 C5GBF2 10286667 IC50 = 200 nM T62431 C9I5TF 10286814 IC50 = 20 nM T62431 CZX24S 10287337 IC50 = 120 nM T62431 C8QH0L 10291291 Ki = 630 nM T62431 C7SFI1 10296883 IC50 > 10000 nM T62431 CZ3BD4 10308373 IC50 = 1100 nM T62431 C08NVH 10308736 IC50 = 78 nM T62431 C3OS2E 10308737 IC50 = 19 nM T62431 C8JQ4V 10309014 IC50 = 500 nM T62431 CK0J9L 10309119 IC50 = 830 nM T62431 COWU64 10309216 IC50 = 850 nM T62431 CK4H8C 10318571 IC50 = 5000 nM T62431 CFN8C2 10343317 IC50 = 50000 nM T62431 CP4M1C 10347718 IC50 > 500000 nM T62431 CC1F4Y 10428841 IC50 = 25000 nM T62431 COW41H 10452792 IC50 = 1500 nM T62431 CC2T0H 10455153 IC50 = 4 nM T62431 C24LNX 10457649 IC50 = 840 nM T62431 CPC6W0 10500718 IC50 = 28000 nM T62431 C62GCM 10504027 IC50 = 45000 nM T62431 CW3F5U 10619651 IC50 = 5000 nM T62431 C1RQ9B 10620637 IC50 = 5000 nM T62431 C0NE7M 10716388 IC50 = 50000 nM T62431 CQGN13 10738302 IC50 = 35000 nM T62431 C2O0WT 10740438 IC50 = 25000 nM T62431 CX36NZ 10761144 IC50 = 5000 nM T62431 C7WYE6 10787405 IC50 = 8000 nM T62431 CDQ43L 10930781 IC50 = 1100 nM T62431 C51SEH 10941165 IC50 = 63000 nM T62431 C04YGB 10995725 IC50 = 71000 nM T62431 CX51GB 10995861 IC50 = 41000 nM T62431 C07EOW 11016822 IC50 = 350000 nM T62431 C2W5RC 11235063 IC50 > 50000 nM T62431 CNBX16 11270660 IC50 > 10000 nM T62431 CMXI90 11324412 Ki = 4 nM T62431 CJC95A 11454205 IC50 > 10000 nM T62431 C0ENJ4 11493171 IC50 = 7610 nM T62431 CC98VE 11501395 IC50 = 4290 nM T62431 COR23C 11523166 IC50 = 23 nM T62431 C4SC3M 11523529 IC50 = 36400 nM T62431 CHX14T 11545405 IC50 = 5360 nM T62431 C26ABY 11551547 IC50 = 7700 nM T62431 CACS26 11561968 Ki > 4000 nM T62431 C9X6EK 11565679 IC50 = 87500 nM T62431 CJO63L 11588347 EC50 = 210 nM T62431 CJE9Z5 11602075 IC50 = 666 nM T62431 C5U4XY 11617275 IC50 = 1186 nM T62431 CYG0Q8 11624063 IC50 = 1570 nM T62431 CK34LS 11632737 IC50 > 50000 nM T62431 CLB7V5 11660668 IC50 = 1100 nM T62431 CAU3O7 11667007 IC50 = 37000 nM T62431 C8XGK5 11667761 IC50 = 22900 nM T62431 CJ9KN7 11683817 IC50 > 10000 nM T62431 C8CMI6 11688688 IC50 = 5620 nM T62431 CU0E8O 11690457 Ki > 4000 nM T62431 CB0AP2 11705863 Ki > 4000 nM T62431 CXM0Q2 11710403 IC50 = 47 nM T62431 C45EWD 11723489 IC50 > 7000 nM T62431 CP7AH3 11755812 IC50 = 50000 nM T62431 C71VOJ 11784504 IC50 = 10 nM T62431 CN1GL0 11838775 IC50 = 3300 nM T62431 CS36BH 11843159 IC50 = 200 nM T62431 COS89C 12017518 IC50 = 150 nM T62431 COIJ48 12968819 IC50 > 500000 nM T62431 C4AIU2 12968822 IC50 > 500000 nM T62431 CLO17Z 15458391 IC50 = 230 nM T62431 CW3RM7 15458392 IC50 = 66 nM T62431 C1B8SF 15603964 EC50 = 9830 nM T62431 C9TU1O 16046126 IC50 > 1000 nM T62431 CKR57M 16086104 IC50 = 1110 nM T62431 C16NRY 16086114 IC50 = 292 nM T62431 CQG45C 16109001 IC50 = 25000 nM T62431 CGC34R 16118737 IC50 > 5000 nM T62431 C5VPH9 16129448 IC50 = 8 nM T62431 CREU56 16201577 IC50 = 100 nM T62431 CQ6G0U 16456747 IC50 = 20000 nM T62431 C0H8UN 16730109 IC50 > 50000 nM T62431 CLWQ98 16744158 IC50 = 3890 nM T62431 C9SVA0 17313189 EC50 = 4140 nM T62431 C9MNP2 17549086 IC50 = 22600 nM T62431 CS85XV 18460827 IC50 = 5000 nM T62431 CN42HV 18460835 IC50 = 2511.89 nM T62431 CJC5F3 20741385 Ki = 82 nM T62431 CK10TP 21029844 EC50 = 290 nM T62431 C5NY4H 21029856 EC50 = 330 nM T62431 CONH43 21106482 IC50 = 1250 nM T62431 C5W9CM 21106492 IC50 = 7665 nM T62431 CL7AB1 21106496 IC50 = 525 nM T62431 CJYA40 22060237 EC50 = 2900 nM T62431 C0L9GZ 22060248 EC50 = 2200 nM T62431 CD45BA 22060262 EC50 = 3400 nM T62431 C9B1PJ 22060268 EC50 = 280 nM T62431 CQ45IN 22060283 EC50 = 4150 nM T62431 CXT9D2 22060303 EC50 = 5800 nM T62431 CD1P0Z 22060450 EC50 = 4250 nM T62431 CA9M7T 22060551 EC50 = 2800 nM T62431 C87GIY 22060633 EC50 = 440 nM T62431 C8V3CB 22060681 EC50 = 670 nM T62431 C7F6WX 22060756 EC50 = 950 nM T62431 C6GWM4 22060878 EC50 = 270 nM T62431 C96JTK 22060949 EC50 = 3100 nM T62431 CP3E1Q 22060990 EC50 = 5080 nM T62431 CMU43A 22061056 EC50 = 900 nM T62431 C5X3AC 22061075 EC50 = 3380 nM T62431 C32ONT 22061080 EC50 = 1730 nM T62431 CQ38IP 22061141 EC50 = 230 nM T62431 CX0T9H 22061183 EC50 = 930 nM T62431 CVMH27 22503663 IC50 > 30 ug.mL-1 T62431 CZ0YD5 22665517 IC50 > 10000 nM T62431 CO15GI 22665531 IC50 > 10000 nM T62431 CA97TZ 22958832 IC50 = 280 nM T62431 CST6I8 22978714 IC50 = 128 nM T62431 C6JV7W 23400934 IC50 > 7000 nM T62431 CD5S7O 23401001 IC50 > 7000 nM T62431 CW7DG1 23467602 IC50 = 17000 nM T62431 CK5N6B 23657635 IC50 = 220 nM T62431 C2S5ZM 23661662 Ki = 41 nM T62431 C3JOC8 24753585 IC50 = 894 nM T62431 C0FI3W 24753683 IC50 = 3020 nM T62431 CFDJ01 24753686 IC50 = 1860 nM T62431 CIZ4V1 24756997 IC50 > 10000 nM T62431 C7YG1N 24759534 IC50 = 440 nM T62431 CLBP72 24798571 IC50 = 2272 nM T62431 C9F1AO 24821023 IC50 > 10000 nM T62431 CC9J2A 24828759 IC50 = 17 nM T62431 CY8L7E 24896769 IC50 > 10000 nM T62431 C5ZM4T 24936119 IC50 > 10000 nM T62431 C4PY9V 25021078 IC50 = 7100 nM T62431 CQ67BO 25113172 IC50 = 6 nM T62431 C36FXD 25138012 IC50 = 26 nM T62431 CP6N4G 25138050 IC50 = 620 nM T62431 CL0Q2A 25138151 IC50 = 7100 nM T62431 CHN12U 25138152 IC50 = 4300 nM T62431 CAU4D5 25138153 IC50 = 230 nM T62431 CID5O7 25169255 Ki = 14 nM T62431 CN2B0H 25169256 IC50 = 26 nM T62431 CWP29U 25242324 IC50 = 371 nM T62431 CC71QJ 27666048 IC50 > 100000 nM T62431 CG9TP5 44187112 IC50 = 4.3 nM T62431 CYSU78 44187114 EC50 = 293 nM T62431 CMC0P7 44188018 IC50 = 64.1 nM T62431 CHJ7G5 44188199 IC50 = 18.6 nM T62431 CI6B2G 44188200 IC50 = 28.3 nM T62431 C9GAR8 44188204 EC50 = 418 nM T62431 C9YP7K 44188382 IC50 = 112 nM T62431 C5XAD9 44188391 EC50 = 251 nM T62431 CO6G9U 44188551 IC50 = 50.2 nM T62431 C43KNU 44189082 EC50 = 643 nM T62431 C8LW9N 44189262 EC50 = 175 nM T62431 C7XBM6 44189444 IC50 = 2.2 nM T62431 C64ZHQ 44189445 EC50 = 270 nM T62431 C2SXL1 44189621 IC50 = 16.5 nM T62431 CQ93BP 44189622 IC50 = 2.6 nM T62431 CRU6J3 44205381 IC50 = 14 nM T62431 C84YBA 44205825 IC50 = 35 nM T62431 C8KNA3 44219632 Ki > 4000 nM T62431 C0VIX4 44219633 Ki > 4000 nM T62431 C58EAY 44280048 IC50 = 160 nM T62431 CQ68RU 44280098 IC50 = 5900 nM T62431 CPED62 44280099 IC50 = 490 nM T62431 CD95UH 44280109 IC50 = 8600 nM T62431 C6T4YW 44280184 IC50 = 1700 nM T62431 C7Z5AR 44280185 IC50 > 30 ug.mL-1 T62431 CK05GC 44280198 IC50 = 3800 nM T62431 C2SUA0 44280286 IC50 = 1600 nM T62431 CT5OS8 44280310 IC50 > 30 ug.mL-1 T62431 C6RWL5 44280317 IC50 = 1500 nM T62431 CKM0S1 44280393 IC50 > 30 ug.mL-1 T62431 CCTV82 44280402 IC50 = 1500 nM T62431 C8HBS5 44280403 IC50 = 3600 nM T62431 CNS2Y3 44280404 IC50 > 30 ug.mL-1 T62431 CY3HS4 44280408 IC50 > 30 ug.mL-1 T62431 CXB92Q 44280462 IC50 = 40000 nM T62431 CINU35 44280484 IC50 = 13000 nM T62431 CQP7R3 44280485 IC50 > 30 ug.mL-1 T62431 C7N0LB 44280690 IC50 = 420 nM T62431 CTU5N8 44280691 IC50 = 71 nM T62431 C8OR3L 44280710 IC50 = 25000 nM T62431 C1RGE3 44315963 IC50 = 171000 nM T62431 CX04DQ 44332978 IC50 = 310000 nM T62431 CDGA70 44335755 IC50 = 678 nM T62431 C0AHT7 44335756 IC50 = 204 nM T62431 CY06LU 44335763 IC50 = 98 nM T62431 C6IGV5 44335771 IC50 = 1000 nM T62431 CLBK94 44335776 IC50 = 60 nM T62431 C0D1KR 44335780 IC50 = 658 nM T62431 CF61IP 44335802 IC50 = 4000 nM T62431 C51AWB 44335814 IC50 = 12 nM T62431 CNZ84V 44335815 IC50 = 100 nM T62431 CR01XF 44335823 IC50 = 8100 nM T62431 C8NAL5 44335826 IC50 = 616 nM T62431 CZ89QH 44335827 IC50 = 133 nM T62431 CHF16Y 44335865 IC50 = 28 nM T62431 CO9K8F 44335885 IC50 = 20 nM T62431 C7Y5ZB 44335902 IC50 = 11 nM T62431 CSJT16 44335920 IC50 = 14 nM T62431 CG05XE 44335921 IC50 = 850 nM T62431 C4WHC0 44336073 IC50 = 465 nM T62431 CVY9W3 44336128 IC50 = 32 nM T62431 C9A2MJ 44336147 IC50 = 273 nM T62431 C1OCP4 44336148 IC50 = 4000 nM T62431 CD9I1Q 44336163 IC50 = 937 nM T62431 C7QZU3 44336168 IC50 = 27 nM T62431 CZ2YC5 44353697 IC50 = 480 nM T62431 C8NBI3 44353815 IC50 = 420000 nM T62431 C8J1NC 44353827 IC50 > 500000 nM T62431 C8FVG3 44353828 IC50 = 389000 nM T62431 CUE3M9 44362038 IC50 = 7700000 nM T62431 C5R4QE 44442729 Ki = 250 nM T62431 CGC76I 44442730 Ki > 10000 nM T62431 CJM6N5 44442731 Ki > 10000 nM T62431 CH2FS6 44442732 Ki > 10000 nM T62431 CZ7FC6 44442733 Ki > 10000 nM T62431 C6PNZ4 44442734 Ki > 10000 nM T62431 C8N1EQ 44442735 Ki > 10000 nM T62431 C26EVP 44442736 Ki = 140 nM T62431 C0S6PN 44442737 Ki = 160 nM T62431 CAZ5O7 44442738 Ki > 10000 nM T62431 CM9XW1 44442739 Ki > 10000 nM T62431 CFOH51 44442740 Ki > 10000 nM T62431 CX10DZ 44442742 Ki = 450 nM T62431 CN12IA 44442744 Ki > 10000 nM T62431 C0DOP6 44442745 Ki = 300 nM T62431 C3VRO9 44557921 IC50 > 10000 nM T62431 CYK76V 44565578 IC50 = 310 nM T62431 CTK09P 44565580 IC50 = 500 nM T62431 C4UF2Y 44565581 IC50 = 616 nM T62431 C6W2HE 44565660 IC50 = 5000 nM T62431 CZT5U3 44565661 IC50 = 8600 nM T62431 CVM07P 44565662 IC50 = 750 nM T62431 C4L1IU 44565681 IC50 = 1 nM T62431 C7JT4S 44565682 IC50 = 1.6 nM T62431 CDQO30 44565695 IC50 = 3.7 nM T62431 C1XGL8 44565696 IC50 = 6 nM T62431 CBAJ92 44565697 IC50 = 7 nM T62431 CW3R6Q 44565698 IC50 = 3600 nM T62431 CU9FS0 44565711 IC50 = 11.2 nM T62431 C7ID3T 44565733 IC50 = 21 nM T62431 C70CWK 44565734 IC50 = 2000 nM T62431 CS5M2E 44565735 IC50 = 2000 nM T62431 C2TOM1 44565736 IC50 = 2000 nM T62431 C6W1KX 44565737 IC50 = 2000 nM T62431 C2B6WH 44565756 IC50 = 53 nM T62431 CF3V9T 44565780 IC50 = 72 nM T62431 CG6QK0 44565781 IC50 = 81 nM T62431 C6F0DP 44565782 IC50 = 92 nM T62431 CVG8M6 44565783 IC50 = 6530 nM T62431 CG56OR 44565801 IC50 = 110 nM T62431 C6G5HC 44565802 IC50 = 120 nM T62431 C1TVM9 44565803 IC50 = 9990 nM T62431 C67APN 44565804 IC50 > 10000 nM T62431 CB36HF 44565843 IC50 = 230 nM T62431 CHR28G 44565867 IC50 = 2.5 nM T62431 C50WBX 44565868 IC50 = 500 nM T62431 C89ILP 44565884 IC50 = 30 nM T62431 C3T7WB 44565885 IC50 = 50 nM T62431 CR2W4L 44565886 IC50 = 500 nM T62431 CB5F4K 44565887 IC50 = 500 nM T62431 CALV38 44565888 IC50 = 500 nM T62431 CAYN97 44588971 IC50 = 1500 nM T62431 CEL6D9 44588972 IC50 = 720 nM T62431 CNZ2H5 44589000 IC50 = 1200 nM T62431 CCYQ91 44589001 IC50 = 6 nM T62431 CV5GD1 44589002 IC50 = 9 nM T62431 C83KEG 44589022 IC50 = 4 nM T62431 CTZX27 44589023 IC50 > 10000 nM T62431 C34KTW 44589024 IC50 = 30 nM T62431 C59BIS 44589025 IC50 = 92 nM T62431 C4TUK3 44589050 IC50 = 30 nM T62431 CNA20V 44589051 IC50 = 6 nM T62431 CA5UF3 44589514 Ki = 33 nM T62431 C3KLD1 44589515 Ki = 50 nM T62431 C7A0UX 44589516 Ki = 23 nM T62431 CYK07V 44589517 Ki = 10 nM T62431 CBV4U7 44590109 IC50 = 5 nM T62431 C5T3IH 44590110 IC50 = 8 nM T62431 C89COX 44590149 Ki = 28 nM T62431 C2BQ4M 44590150 Ki = 44 nM T62431 C6NB9K 44590204 Ki = 23 nM T62431 CQ0NU8 44590205 Ki = 10 nM T62431 COY57J 44592504 IC50 = 25000 nM T62431 C87MBD 44593467 IC50 = 1000 nM T62431 C2PX5O 44593468 IC50 = 1817 nM T62431 CZ20KC 44593469 IC50 = 22 nM T62431 CM3T7B 44593470 IC50 = 32 nM T62431 CD2FE4 44593471 Ki = 56 nM T62431 CS8GE3 44593472 IC50 = 110 nM T62431 CKM4H0 44593475 IC50 = 9 nM T62431 CU3RF1 45139989 IC50 > 10000 nM T62431 CQGZ06 45139991 IC50 > 10000 nM T62431 CY83PR 45267327 IC50 > 1000 nM T62431 C84QFJ 45269074 IC50 = 300 nM T62431 C2JVA4 45270368 IC50 = 80 nM T62431 C3DH8I 45273358 IC50 > 1000 nM T62431 CET79H 45493316 IC50 = 12000 nM T62431 CZGB46 46180666 IC50 > 1000 nM T62431 CZ58FY 46215814 IC50 = 4000 nM T62431 CY3HW5 46224684 IC50 > 10000 nM T62431 C7ON5A 46233287 IC50 > 10000 nM T62431 C67UQY 46234933 EC50 = 2366 nM T62431 C64RIB 46325413 IC50 = 9900 nM T62431 CGI8Z7 46337935 IC50 = 28000 nM T62431 CC2O9R 46865656 IC50 = 31.62 nM T62431 CLS29B 46872626 IC50 > 10000 nM T62431 C9L3XR 49838879 IC50 > 50000 nM T62431 CF91RS 49843531 IC50 > 10000 nM T62431 C2Y6QS 50938552 IC50 > 10000 nM T62431 C9NYP4 51036677 IC50 > 10000 nM T62431 C4WRY3 51037112 IC50 > 10000 nM T62431 CRI28Z 51037948 IC50 > 10000 nM T62431 CM24LF 52938983 IC50 < 1 nM T62431 C0AU2P 53207882 IC50 = 30000 nM T62431 CR36JQ 53232414 IC50 = 2.3 nM T62431 C1K8ZJ 53232523 IC50 = 1.9 nM T62431 CS8I3Y 53232528 IC50 = 307 nM T62431 CJP9Q0 53242134 IC50 = 0.9 nM T62431 CX21TF 53250672 IC50 = 0.8 nM T62431 CAB3J0 53250673 IC50 = 0.5 nM T62431 CZ9V8X 53251797 EC50 = 35 nM T62431 CR37YZ 53251953 IC50 = 4.7 nM T62431 CL80MF 53252274 EC50 = 9 nM T62431 CNPM14 53341082 IC50 > 3000 nM T62431 C8NA4L 53384644 IC50 > 30000 nM T62431 CY8WL1 54586678 IC50 = 850 nM T62431 CN9QD7 56643097 IC50 > 10000 nM T62431 CVG04B 56659303 IC50 = 25.12 nM T62431 CRTE61 56659304 IC50 = 125.89 nM T62431 C3R8ZJ 56659305 IC50 = 3981.07 nM T62431 CD64XI 56664830 IC50 = 570000 nM T62431 CUD91I 56664831 IC50 = 1200 nM T62431 C6B7WR 56666236 IC50 = 398.11 nM T62431 CVBA49 56666237 IC50 = 1258.93 nM T62431 C45XIM 56666238 IC50 = 125.89 nM T62431 C5OF9G 56669642 IC50 = 12.59 nM T62431 CUP61N 56671791 IC50 = 79.43 nM T62431 C6E7WM 56673153 IC50 = 398.11 nM T62431 C2Z1LP 56673154 IC50 = 1258.93 nM T62431 CT0C2N 56675134 IC50 = 62000 nM T62431 CF3G7P 56676480 IC50 = 501.19 nM T62431 CN4US8 56676481 IC50 = 100 nM T62431 C49LUC 56676482 IC50 = 10 nM T62431 CP14LU 56678505 IC50 = 125.89 nM T62431 CDS09F 56679795 IC50 = 79.43 nM T62431 CU04BI 56679796 IC50 = 398.11 nM T62431 CTEK36 56679797 IC50 = 3.981 nM T62431 CZSM95 57412684 IC50 > 10000 nM T62431 CDC4I7 57856403 EC50 = 248 nM T62431 CME1I7 57856413 IC50 = 466 nM T62431 C8GIZ4 57856426 IC50 = 1.5 nM T62431 C3VM8D 57856427 IC50 = 37.4 nM T62431 C3LPO7 58317600 IC50 = 3.1 nM T62431 CDB42N 58513640 IC50 = 5.7 nM T62431 C16CEO 58513660 IC50 = 17.8 nM T62431 C4WMF1 58513688 IC50 = 377 nM T62431 CT3EW2 59292007 IC50 > 1000 nM T62431 CG2R6C 59473104 IC50 = 2.1 nM T62431 CCEB81 59473148 EC50 = 15 nM T62431 C9QYR7 59473155 IC50 = 8.5 nM T62431 CXUH63 59473230 IC50 = 6.3 nM T62431 CB68MW 59473263 IC50 = 2.3 nM T62431 CJ4WU7 59473266 IC50 = 2.7 nM T62431 C9GC4O 59473273 IC50 = 7 nM T62431 C6P8FT 59473280 EC50 = 80 nM T62431 CRG50X 59473315 IC50 = 20.9 nM T62431 C0JKO7 59473380 EC50 = 24 nM T62431 CM4RT7 59473397 EC50 = 86 nM T62431 CACJ63 59473411 IC50 = 10.4 nM T62431 CTG92P 59473462 IC50 = 4.7 nM T62431 C5G7MI 59473523 EC50 = 151 nM T62431 CCK7W1 59473555 IC50 = 23.1 nM T62431 CD6ZP4 59473598 IC50 = 7.6 nM T62431 CD8A3W 59473640 IC50 = 0.44 nM T62431 CD2O3Z 59473650 IC50 = 12.3 nM T62431 CS49QD 59473651 EC50 = 168 nM T62431 CXJ63M 59603829 IC50 = 750 nM T62431 CQEU96 59603842 IC50 = 42 nM T62431 COH62U 60097413 IC50 > 2500 nM T62431 C1MR8Q 60097495 IC50 > 2500 nM T62431 CL4G2M 60147015 IC50 = 100 nM T62431 C3PQE0 60147016 IC50 = 2 nM T62431 CTO6J5 60203901 IC50 = 7 nM T62431 C2SR0W 64008775 IC50 = 50118.72 nM T62431 CPR43N 66550117 IC50 = 93 nM T62431 CZ2PY6 66551542 IC50 = 47 nM T62431 C6TN4K 66551543 IC50 = 423 nM T62431 C8CI6S 66551544 IC50 = 50 nM T62431 CA42UL 66554658 IC50 = 79.43 nM T62431 CX25QN 66555696 IC50 = 125.89 nM T62431 CL0X8S 66555697 IC50 = 158.49 nM T62431 C2Y7FX 66555698 IC50 = 15.85 nM T62431 C8PST7 66556032 IC50 = 3.981 nM T62431 CV8JO4 66556033 IC50 = 39.81 nM T62431 CSZ6I5 66556035 IC50 = 63.1 nM T62431 C6SL1Q 66556036 IC50 = 63.1 nM T62431 CX6J3B 66556201 IC50 = 5.012 nM T62431 CHWG72 66556203 IC50 = 50.12 nM T62431 CVPT78 66556206 IC50 = 6309.57 nM T62431 C0F5HW 66556207 IC50 > 25118.86 nM T62431 C6E7CU 66556365 IC50 = 25.12 nM T62431 CR7JT9 66556366 IC50 = 199.53 nM T62431 CSM89V 66556371 IC50 = 1000 nM T62431 CK9QI1 66556533 IC50 = 63.1 nM T62431 CA1Z4Q 66556534 IC50 = 251.19 nM T62431 CNRZ13 66556535 IC50 = 50.12 nM T62431 C7MD5X 66556536 IC50 = 251.19 nM T62431 C01RFU 66556542 IC50 = 25.12 nM T62431 C1HSE0 67035086 IC50 > 10000 nM T62431 CWI6K5 67035106 IC50 > 10000 nM T62431 C38RGB 67035556 IC50 > 10000 nM T62431 C8B0LN 67129951 EC50 = 346 nM T62431 C37NKO 67129970 IC50 = 97 nM T62431 CK80LJ 67130050 EC50 = 34 nM T62431 CV63UL 67240318 IC50 > 10000 nM T62431 COM54X 67775149 IC50 = 19 nM T62431 C4M9LX 68289700 IC50 = 158.49 nM T62431 C07JAL 68290083 IC50 = 398.11 nM T62431 CC70KY 68290508 IC50 = 100 nM T62431 C8I7GC 68293638 IC50 > 10000 nM T62431 CD56XK 68293660 IC50 > 10000 nM T62431 CIB52Q 68309298 IC50 = 316.23 nM T62431 CBGL83 68309299 IC50 = 31.62 nM T62431 CWDS89 68310172 IC50 = 100 nM T62431 C6TJF9 68751510 IC50 = 179 nM T62431 C7GRV2 68755406 IC50 = 61 nM T62431 C0HA8V 68783839 IC50 = 44 nM T62431 C5ZC4A 69000930 EC50 = 244 nM T62431 CHWF15 69002997 IC50 = 17.7 nM T62431 C3BE1J 70664916 IC50 = 398.11 nM T62431 C1BP3M 70665059 IC50 = 39.81 nM T62431 C5SR8C 70665106 IC50 = 199.53 nM T62431 CDF8I5 70665119 IC50 = 3162.28 nM T62431 C4U2GE 70665128 IC50 = 63.1 nM T62431 CULR51 70665234 IC50 = 100 nM T62431 C1AN6J 70665241 IC50 = 79.43 nM T62431 C8RB5N 70665321 IC50 = 158.49 nM T62431 CDA14G 70665372 IC50 = 1995.26 nM T62431 C6S8CL 70665375 IC50 = 251.19 nM T62431 CH7O9I 70665379 IC50 = 630.96 nM T62431 CB2Y9Z 70665386 IC50 = 199.53 nM T62431 CSG04B 70665393 IC50 = 316.23 nM T62431 CXCW07 70665412 IC50 = 39.81 nM T62431 CE39KJ 70680736 IC50 = 47 nM T62431 C6U2WZ 70687578 IC50 = 20 nM T62431 CDI9F6 70981182 IC50 > 10000 nM T62431 C8JL2S 71074152 IC50 = 3 nM T62431 CZ29NF 71113911 IC50 = 25.12 nM T62431 CT1L2V 71113915 IC50 = 199.53 nM T62431 CYLA18 71279311 IC50 = 34 nM T62431 C47QTF 71279423 IC50 = 5 nM T62431 CH4T8Z 71279444 IC50 = 7 nM T62431 C2YHK4 71279453 IC50 = 5 nM T62431 C4E1RT 71279494 IC50 = 61 nM T62431 CZR37K 71279507 IC50 = 78 nM T62431 CU4P3X 71279543 IC50 = 5 nM T62431 C5L8SW 71279563 IC50 = 4 nM T62431 CQ7L0A 71279608 IC50 = 88 nM T62431 CV96FO 71279672 IC50 = 2 nM T62431 CKJ58I 71279693 IC50 = 19 nM T62431 C6RHS3 71279723 IC50 = 129 nM T62431 C7KQZ0 71279846 IC50 = 3 nM T62431 CZY5P7 71279859 IC50 = 4 nM T62431 C42LGQ 71279939 IC50 = 36 nM T62431 CXZG59 71280008 IC50 = 26 nM T62431 C5TXH9 71280067 IC50 = 4 nM T62431 CW0FK6 71280128 IC50 = 68 nM T62431 CEO08K 71280143 IC50 = 64 nM T62431 CGI01S 71280152 IC50 = 195 nM T62431 C5IS6H 71280272 IC50 = 4 nM T62431 C61BWN 71280407 IC50 = 10 nM T62431 C5CTH0 71280416 IC50 = 5 nM T62431 CWV13N 71280420 IC50 = 738 nM T62431 CHY7N4 71280456 IC50 = 1 nM T62431 C63EIL 71280539 IC50 = 3 nM T62431 CUP25C 71280634 IC50 = 30 nM T62431 C3LOB1 71285746 IC50 = 47 nM T62431 C0GXY1 71287917 IC50 = 13 nM T62431 C4AP9F 71288434 IC50 = 19 nM T62431 CXU4Q3 71288435 IC50 = 132 nM T62431 C68LPJ 71288456 IC50 = 6 nM T62431 CTS5B4 71288807 IC50 = 68 nM T62431 CB5MS7 71288819 IC50 = 135 nM T62431 C1W5VU 71451822 IC50 = 406 nM T62431 CGL6Q7 71451823 IC50 = 25 nM T62431 CW29RV 71457142 IC50 = 1 nM T62431 CC6D7U 71459019 IC50 = 351 nM T62431 CTJX41 71460808 IC50 = 127 nM T62431 CR8OA2 71462533 IC50 = 16 nM T62431 C9DIK2 71512060 IC50 > 10000 nM T62431 C5RB1A 71522868 IC50 = 2.8 nM T62431 CYU96B 71522956 IC50 < 1.5 nM T62431 CL1AC3 71523041 IC50 < 1.5 nM T62431 C3J7MC 71523042 IC50 < 1.5 nM T62431 C5K9GY 71523123 IC50 < 1.5 nM T62431 C1M3ET 71523125 IC50 > 1.5 nM T62431 CI71DK 71533675 IC50 = 0.06 nM T62431 CRO3H4 71544435 IC50 = 19 nM T62431 C2PC6S 71547342 IC50 = 0.1 nM T62431 CP38KG 71547422 IC50 = 0.1 nM T62431 CD97ZU 71547584 IC50 = 0.8 nM T62431 CIRZ76 71547586 IC50 = 0.5 nM T62431 CCN01X 71547862 IC50 > 10000 nM T62431 CC0B1F 71547911 IC50 = 9 nM T62431 CEV53L 71548006 IC50 = 0.6 nM T62431 CRX81Q 71575642 IC50 > 10000 nM T62431 CH5LE3 71598532 IC50 = 3.162 nM T62431 C5IKR3 71625970 IC50 = 3.162 nM T62431 CC54ZM 71625972 IC50 = 398.11 nM T62431 C09VQL 71625973 IC50 = 251.19 nM T62431 C5NA4Y 71625975 IC50 = 199.53 nM T62431 CW7DI6 71626041 IC50 = 10 nM T62431 CGR3I5 71626043 IC50 = 10 nM T62431 CCQ69B 71626102 IC50 = 3.162 nM T62431 CEPZ57 71626162 IC50 = 63.1 nM T62431 C2AU1I 71626163 IC50 = 158.49 nM T62431 C2WJX0 71626755 IC50 = 10 nM T62431 CTRE28 71626822 IC50 = 3.981 nM T62431 C8TID3 71626894 IC50 = 199.53 nM T62431 C26TXG 71626895 IC50 = 25.12 nM T62431 C4DHC9 71626896 IC50 = 31.62 nM T62431 CJV92N 71626898 IC50 = 158.49 nM T62431 C3XV8I 71626968 IC50 = 3.981 nM T62431 C7GZI2 71626969 IC50 = 39.81 nM T62431 CX0VE7 71626971 IC50 = 251.19 nM T62431 C5LT9M 71698375 IC50 = 36.6 nM T62431 CS62NH 71698376 IC50 = 1 nM T62431 CVDL37 71698378 IC50 = 0.7 nM T62431 CI8X1R 71698379 IC50 = 1.7 nM T62431 C6L7SX 71698642 IC50 = 19.5 nM T62431 CTW95M 71698643 IC50 = 0.7 nM T62431 CY10TN 71698644 IC50 = 8 nM T62431 CTNS87 71698733 IC50 = 20.4 nM T62431 CS8CZ7 71718968 IC50 = 563 nM T62431 CPNI04 71842879 IC50 = 3200 nM T62431 CKMZ39 72202597 IC50 = 99 nM T62431 CO5XJ3 72202738 IC50 = 14 nM T62431 CJTS50 72202874 IC50 = 5 nM T62431 CCT15O 72703033 IC50 = 5 nM T62431 C95XRF 73352323 IC50 = 937 nM T62431 CHV7Q0 73356064 IC50 = 130 nM T62431 CO6I7Q 73777147 IC50 = 630.96 nM T62431 CO0LS1 73777169 IC50 > 50118.72 nM T62431 CGC10B 73777172 IC50 = 199.53 nM T62431 C5LPC2 73777186 IC50 = 501.19 nM T62431 C3NDE7 73777188 IC50 = 10 nM T62431 CS71JA 73777210 IC50 = 39.81 nM T62431 CK3W5O 73777215 IC50 = 39.81 nM T62431 CENQ80 73777235 IC50 = 25.12 nM T62431 CG6T5S 76072368 IC50 = 49.8 nM T62431 CZ97VP 86294733 IC50 = 22 nM T62431 CPG3A5 86302574 IC50 > 30000 nM T62431 CXJA65 86685547 IC50 = 1 nM T62431 CWMX37 87228576 IC50 = 6.3 nM T62431 CGY2Z5 89486768 IC50 = 0.8 nM T62431 CS7GX8 89708625 IC50 = 1 nM T62431 C1HW4B 89735655 IC50 = 12000 nM T62431 C5LQG9 89769061 IC50 = 100 nM T62431 C4KGB3 89845254 IC50 = 9.2 nM T62431 C1T7AE 89845281 IC50 = 326 nM T62431 CN6H0G 89846362 IC50 = 22.8 nM T62431 CN76VK 89912923 IC50 = 1000 nM T62431 C9UZX2 90355303 IC50 = 0.5 nM T62431 CY0UC4 90645194 IC50 > 10000 nM T62431 CV9H8U 90656285 IC50 = 1 nM T62431 CG7E1U 90656286 IC50 = 4 nM T62431 CDF9O2 90656287 IC50 = 3 nM T62431 CB4D0X 90656289 IC50 = 1900 nM T62431 C2YHC1 90656832 IC50 = 26.8 nM T62431 C12SAH 90656833 IC50 = 65 nM T62431 CF89DA 90664659 IC50 = 41 nM T62431 CUCS06 91885526 IC50 = 5 nM T62431 CACB62 91885527 IC50 = 166 nM T62431 CCVL49 100942265 IC50 = 434000 nM T62431 CU6ZJ3 102515519 IC50 = 11.5 nM T62431 CK4Z3C 102515520 IC50 = 7.3 nM T62431 CEPI85 102532139 IC50 = 0.5 nM T62431 CG1R8H 102532140 IC50 = 2.5 nM T62431 C1TF9K 118368174 IC50 = 0.7 nM T62431 CZ68JM 118368188 IC50 = 5 nM T62431 C1GI7A 118372967 IC50 = 530 nM T62431 CY7BI2 118706214 IC50 > 10000 nM T62431 CHT6K9 118728811 Ki > 4000 nM T62431 CUA3Y2 118728812 Ki > 4000 nM T62431 CDQ78G 118728813 Ki > 4000 nM T62431 CZ6XL7 118728814 Ki > 4000 nM T62431 CMO67K 118728815 Ki > 4000 nM T62431 CR2M0Q 118728816 Ki > 4000 nM T62431 C62SCL 118728817 Ki > 4000 nM T62431 CSB30C 118728819 Ki > 4000 nM T62431 CV7XU8 118728820 Ki = 3400 nM T62431 C3J1EX 118728821 Ki > 4000 nM T62431 CIWB78 118728822 Ki > 4000 nM T62431 CP18SE 118728823 Ki > 4000 nM T62431 CM42CA 118728824 Ki > 4000 nM T62431 C9Q7CL 118728825 Ki > 4000 nM T62431 CCR3S0 118728826 Ki > 4000 nM T62431 CK2R8V 118729093 EC50 = 380 nM T62431 CBV7U9 118729096 EC50 = 370 nM T62431 CVP1Q7 118729097 EC50 = 430 nM T62431 C13FOT 118729098 EC50 = 940 nM T62431 C5VJ2X 118729099 EC50 = 440 nM T62431 C3N1PM 118729100 EC50 = 490 nM T62431 CI8L3H 118729102 EC50 = 760 nM T62431 CY8WK7 118729103 EC50 = 530 nM T62431 CKCY70 118729104 EC50 = 450 nM T62431 CG5MR2 118729105 EC50 = 1550 nM T62431 C0EUI4 118729106 EC50 = 430 nM T62431 CXD3H4 118729107 EC50 = 1100 nM T62431 CUK5M0 118729108 EC50 = 400 nM T62431 CEM5Q6 118729109 EC50 = 210 nM T62431 C0BWF7 118729110 EC50 = 1290 nM T62431 CSL78U 118731592 IC50 = 2958 nM T62431 C3EK8F 118731593 IC50 = 1130 nM T62431 CCV52L 118731594 IC50 = 326 nM T62431 C6M1AQ 118731595 IC50 = 13 nM T62431 CN75IB 118733346 IC50 = 8.8 nM T62431 CC2I1K 118733347 IC50 = 7 nM T62431 C1AVK5 118733348 IC50 = 371 nM T62431 C43XUF 118733349 IC50 = 184 nM T62431 C7XG3O 118733350 IC50 = 5 nM T62431 CNYV64 118733351 IC50 = 0.1 nM T62431 CLI96Y 118733352 IC50 = 0.9 nM T62431 C5Q2VW 118733353 IC50 = 0.2 nM T62431 C5YB6G 118733354 IC50 = 0.01 nM T62431 C5OQ3B 118733356 IC50 = 51 nM T62431 C7NJE0 118733357 IC50 = 60 nM T62431 C32NYW 118733358 IC50 = 0.4 nM T62431 CC0W7L 118733359 IC50 = 1 nM T62431 C7K2MN 118733360 IC50 = 2 nM T62431 C2Y7MH 118733361 IC50 = 7 nM T62431 CRO7S5 118733755 IC50 = 165 nM T62431 C2XZN0 118733756 IC50 = 170 nM T62431 CZ17EX 121269180 IC50 = 6.2 nM T62431 CG9Q1H 121320416 IC50 = 153000 nM T62431 C08KEM 122179540 IC50 = 4000 nM T62431 CG0RP7 122179547 IC50 = 4400 nM T62431 C1A0SQ 122179548 IC50 = 7900 nM T62431 C5AFZ6 122191639 IC50 = 38 nM T62431 CW5SL7 122191640 IC50 = 89 nM T62431 CT5B0E 122191641 IC50 = 538 nM T62431 CTX98S 122191642 IC50 = 46 nM T62431 CEK1V4 122191643 IC50 = 247 nM T62431 CY21TW 122191644 IC50 = 57 nM T62431 CIR25H 122191977 IC50 = 16 nM T62431 CFG87R 122191978 IC50 = 107 nM T62431 CW4S2I 122192139 IC50 = 871 nM T62431 C8KN5P 122192140 IC50 = 5.4 nM T62431 CH0PT3 122192141 IC50 = 38 nM T62431 C28KRS 122192142 IC50 = 3.5 nM T62431 C23GHM 122192143 IC50 = 71.8 nM T62431 CXG12E 122192144 IC50 = 39.1 nM T62431 C1RG4Z 122192145 IC50 = 3.7 nM T62431 C8ICQ1 122192146 IC50 = 13.2 nM T62431 CUEF56 122192147 IC50 = 5 nM T62431 C2JN3R 122192148 IC50 = 17.3 nM T62431 CJI49C 122192149 IC50 = 7.3 nM T62431 CXM27E 122192150 IC50 = 14.4 nM T62431 CHT1C3 122192151 IC50 = 8.9 nM T62431 C1Q8SU 122192152 IC50 = 7.9 nM T62431 CZ6V4R 122192153 IC50 = 61.4 nM T62431 CO1J7B 122192154 IC50 = 100.8 nM T62431 CBX83N 122192155 IC50 = 144.5 nM T62431 CC7V2M 122192156 IC50 = 5994 nM T62431 C4X7SD 122192466 IC50 > 10000 nM T62431 CUO0C5 132156633 IC50 > 10000 nM T62431 CQF12X 134138313 IC50 = 24 nM T62431 CU3G0M 134141942 IC50 = 990 nM T62431 CK8R5Y 134145931 IC50 = 7 nM T62431 CD5MT9 134146337 IC50 = 2.3 nM T62431 CPQ7C5 134148481 IC50 = 1600 nM T62431 CB09CT 134152904 IC50 > 10000 nM T62431 CEU8B2 134154976 IC50 = 9 nM T62431 C2AN7T 134611886 IC50 > 100000 nM T62431 CZ2RP8 134817809 IC50 = 3162.28 nM T62431 C54FXD 134957362 IC50 > 10000 nM T62431 CMD98Q 135399658 IC50 = 2520 nM T62431 C5L3AB 135408347 IC50 = 17000 nM T62431 CPZ93E 135437725 IC50 = 4000 nM T62431 CRY3K8 135456003 IC50 > 20000 nM T62431 C86WCU 135469510 IC50 > 20000 nM T62431 CQS0J5 135494737 IC50 = 40000 nM T62431 CPQB94 135498616 IC50 = 24000 nM T62431 CTQ37F 135510931 IC50 = 30900 nM T62431 CTJ48K 135524085 IC50 = 2500 nM T62431 CUT1W7 135524168 IC50 = 6200 nM T62431 C4SN0G 135548971 IC50 = 168000 nM T62431 CY4D8I 135566504 Ki = 351.4 nM T62431 CJ03PU 135566610 IC50 = 286.9 nM T62431 CQ9A5I 135566611 IC50 = 938.6 nM T62431 C42TOW 135566612 IC50 = 358.2 nM T62431 CN48IF 135566613 IC50 = 2469 nM T62431 CIS2L5 135566617 IC50 = 8 nM T62431 C67IYS 135566618 IC50 = 4 nM T62431 CI47VJ 135566923 IC50 = 4 nM T62431 CHU3A2 135635724 IC50 = 26000 nM T62431 CPV59N 135685787 Ki > 4000 nM T62431 C29PWN 135886762 IC50 = 18400 nM T62431 CG3UZ1 135927974 Ki > 1000 nM T62431 CF1PS8 135934877 Ki = 690 nM T62431 CTRL59 135976660 Ki = 1800 nM T62431 CHA4N2 136013680 IC50 > 10 nM T62431 CP5SD0 136016241 IC50 = 185.6 nM T62431 CJ9B4L 136036267 IC50 = 500 nM T62431 CHL5Z7 136056540 IC50 = 5 nM T62431 CO0L9T 136056541 IC50 = 2 nM T62431 CLIE18 136056542 IC50 = 320 nM T62431 CM7V8J 136056543 IC50 = 1600 nM T62431 C64BEV 136056544 IC50 = 322 nM T62431 CP1MX4 136056545 IC50 = 232 nM T62431 C4AR8N 136056546 IC50 = 209 nM T62431 CC10GD 136056547 IC50 = 165 nM T62431 CN1PY3 136056548 IC50 = 299 nM T62431 CI8Y0U 136056549 IC50 = 480 nM T62431 CQ84IZ 136180335 Ki > 4000 nM T62431 C1YUD0 136219394 IC50 > 10 nM T62431 CIU8W3 136254389 IC50 > 10 nM T62431 CH0B9N 136499039 IC50 = 11.7 nM T62431 CCA91J 137632410 EC50 = 30 nM T62431 CI1E8V 137634241 IC50 = 7 nM T62431 CO02IV 137637220 IC50 = 1370 nM T62431 C4TFB1 137638523 IC50 = 12 nM T62431 CZHW58 137644151 IC50 = 47 nM T62431 C7ZX6K 137644496 EC50 = 18 nM T62431 CQC3D4 137644670 IC50 = 63 nM T62431 C8O7WF 137645333 EC50 = 43 nM T62431 CCIM31 137647884 IC50 = 20 nM T62431 CU0J4C 137650753 IC50 = 41 nM T62431 CTM95K 137654359 EC50 = 49 nM T62431 CSU12F 137655385 IC50 = 6 nM T62431 CTQA98 137659595 IC50 = 13 nM T62431 CQS10B 137662049 IC50 = 5 nM T62431 CO7Y6G 145966466 IC50 > 10000 nM T62431 CA5T8S 145966795 IC50 > 10000 nM T62431 CTJE41 145966905 IC50 > 10000 nM T62431 CJB41K 145973790 IC50 = 360 nM T62431 C1E0IL 145975398 IC50 > 10000 nM T62431 C9YO2G 145979014 IC50 = 3162.28 nM T62431 C3LIQ9 145979139 IC50 = 1258.93 nM T62431 C10NKS 145979484 IC50 = 794.33 nM T62431 C4LI0Z 145980781 IC50 = 3162.28 nM T62431 C6O9QR 145980932 IC50 = 12589.25 nM T62431 CT6V8J 145980993 IC50 = 1000 nM T62431 C71HNZ 145981987 IC50 = 158.49 nM T62431 CSM3O1 145982265 IC50 = 398.11 nM T62431 C06SXC 145982472 IC50 = 3162.28 nM T62431 C17DUW 145984656 IC50 = 12589.25 nM T62431 C1Z7EV 145985173 IC50 = 1584.89 nM T62431 CA1H6N 145986412 IC50 > 25118.86 nM T62431 CQ0OU9 145986469 IC50 = 1584.89 nM T62431 CU9N0L 145986557 IC50 > 25118.86 nM T62431 CF81XA 145987230 IC50 = 3162.28 nM T62431 CK72YJ 145987295 IC50 = 1995.26 nM T62431 CL3GH2 145987616 IC50 = 3162.28 nM T62431 C1K3SM 145988260 IC50 = 3162.28 nM T62431 CL98WX 145988953 IC50 = 3162.28 nM T62431 CL68AC 145989230 IC50 = 2511.89 nM T62431 C83WRP 145989694 IC50 > 25118.86 nM T62431 CA19KT 145989776 IC50 = 3162.28 nM T62431 C6ISX4 145989906 IC50 = 398.11 nM T62431 C5SP6O 145990231 IC50 = 2511.89 nM T62431 CK46XM 145990305 IC50 = 794.33 nM T62431 C1I5ZT 145991436 IC50 = 3162.28 nM T62431 C9ZL6B 145991873 IC50 = 12589.25 nM T62431 C4RKM8 145992180 IC50 = 3162.28 nM T62431 CN5AK8 145992304 IC50 = 2511.89 nM T62431 CGTE60 145992840 IC50 > 25118.86 nM T62431 CMZ81J 145993911 IC50 = 5011.87 nM T62431 C2MD1Q 155513187 IC50 > 10000 nM T62431 CZEO50 155513953 IC50 = 3.981 nM T62431 CM0IC7 155521232 IC50 = 158.49 nM T62431 C2EHI7 155524928 IC50 = 19.95 nM T62431 C0DZ9X 155527985 IC50 = 2.512 nM T62431 CFR56S 155533031 IC50 = 7.943 nM T62431 C9JD7A 155535968 IC50 = 6.31 nM T62431 C2CG1A 155537016 IC50 > 10000 nM T62431 CTSM92 155538441 IC50 = 5.1 nM T62431 CF1AJ2 155544000 IC50 = 79.43 nM T62431 CIY5U0 155556737 IC50 = 31.62 nM T62431 COSE65 155561444 IC50 = 199.53 nM T62431 D00EIL 6419747 IC50 = 14 nM T62431 D00RIX 5280443 EC50 = 3000 nM T62431 D03OKV 9844320 IC50 > 10000 nM T62431 D04PEI 11467730 IC50 > 50000 nM T62431 D04TLI 23657507 IC50 = 4 nM T62431 D06HVH 54613583 IC50 > 10000 nM T62431 D06WGX 9549184 IC50 > 25000 nM T62431 D07ADX 54764565 IC50 = 731 nM T62431 D08HFG 24809764 IC50 > 10000 nM T62431 D09HVH 135566652 IC50 > 10 nM T62431 D09KEB 11493841 IC50 = 5 nM T62431 D0C7AS 10593843 IC50 = 18000 nM T62431 D0D6MH 11617559 IC50 > 16000 nM T62431 D0EU1R 46215815 IC50 > 25118 nM T62431 D0F0VD 135465539 IC50 > 20000 nM T62431 D0GN5Z 5281295 IC50 = 4630 nM T62431 D0J3LR 11634725 Ki > 4000 nM T62431 D0L1PW 9904854 Ki = 96 nM T62431 D0L4WN 31420 IC50 > 40000 nM T62431 D0MF5Y 5281614 IC50 = 15000 nM T62431 D0NJ4H 5281670 IC50 = 28000 nM T62431 D0O0VZ 667639 IC50 = 5 ug.mL-1 T62431 D0O9UR 638439 IC50 = 76000 nM T62431 D0OZ2S 11785878 IC50 = 200 nM T62431 D0Q3EW 9549303 IC50 = 887 nM T62431 D0Q3GG 667601 IC50 = 38000 nM T62431 D0R7BX 75791 IC50 = 12000000 nM T62431 D0T2NE 58056092 IC50 = 410 nM T62431 D0T3PW 5281672 EC50 = 54000 nM T62431 D0T4MJ 9549296 IC50 = 41 nM T62431 D0X7IM 7595 IC50 > 660000 nM T61744 D05MQK 110635 IC50 > 10000 nM T61744 D09QEI 4740 IC50 = 168000 nM T61744 D0NJ3V 4680 IC50 = 1600 nM T61744 D0R4UW 449193 IC50 = 0.35 nM T61744 D0R6RC 54675777 IC50 = 100000 nM T61744 D0Z7ZM 135398744 IC50 = 5000 nM T61744 D00XVL 42639643 Ki = 62 nM T61744 D03QJL 3671 IC50 = 54 nM T61744 D09TFB 9896267 IC50 = 23 nM T61744 D0M7CB 9919680 IC50 = 5.1 nM T61744 D0SM0W 44591583 IC50 = 55 nM T61744 D0T5PO 5092 IC50 = 10.7 nM T61744 D0Z2FB 154575 IC50 = 1.6 nM T61744 D00YPW 135399235 Ki > 50000 nM T61744 D02EMR 151170 IC50 = 38 nM T61744 D07FHZ 5087 EC50 = 3300 nM T61744 D08SNX 135430158 Ki = 3900 nM T61744 D0BK6B 3021729 Ki > 50000 nM T61744 D0C5PA 183812 IC50 = 38 nM T61744 D0D2PQ 9953237 IC50 = 68 nM T61744 D0K2BQ 71356 EC50 = 910 nM T61744 D0UG4T 127928 Ki = 4 nM T61744 C68GUT 36755 IC50 = 245 nM T61744 COFE25 70387 IC50 > 10000 nM T61744 C4B3YS 78864 IC50 = 162 nM T61744 C1B6ZL 662965 IC50 = 24 nM T61744 C0T7WK 3071941 IC50 = 0.6 nM T61744 C69BNV 3261457 IC50 = 22 nM T61744 CX84RI 3548051 IC50 = 95 nM T61744 CHV64Q 3713518 IC50 = 63 nM T61744 CL1Q4X 4254532 IC50 = 48 nM T61744 C4LDN3 5136241 Ki = 66000 nM T61744 CZ60QE 6501454 Ki = 131000 nM T61744 CJPQ16 6603746 IC50 = 4300 nM T61744 C0XDR3 7447730 Ki = 115000 nM T61744 CFJ62Y 9799389 EC50 = 250 nM T61744 CZH08Y 9802738 IC50 > 10000 nM T61744 CWGO48 9808563 EC50 = 220 nM T61744 CYXD04 9810934 IC50 = 11 nM T61744 CZV60D 9825288 IC50 = 1.2 nM T61744 C97VAE 9825776 IC50 = 35 nM T61744 C27NGI 9827594 IC50 = 6 nM T61744 CUJN41 9828771 IC50 = 1 nM T61744 C95MZB 9829952 IC50 = 0.8 nM T61744 CL70YN 9840066 IC50 = 2.2 nM T61744 C9XY6D 9849838 IC50 = 0.6 nM T61744 C6KRA9 9850032 IC50 = 1.2 nM T61744 CF78JT 9850277 IC50 = 0.8 nM T61744 CAY84B 9869820 IC50 = 0.85 nM T61744 CU4R5A 9884190 EC50 = 15 nM T61744 C3X9JB 9885877 IC50 = 17.5 nM T61744 CCGB72 9915714 IC50 = 0.8 nM T61744 C6YED1 9916317 IC50 = 2.4 nM T61744 C4UM2G 9916436 IC50 = 1.3 nM T61744 C76RTB 9924539 IC50 = 123 nM T61744 C81LSK 9928390 IC50 = 140 nM T61744 C1F4WB 9932192 IC50 = 0.37 nM T61744 CBO5M8 9936981 IC50 = 6 nM T61744 C40NIG 9938153 IC50 = 8 nM T61744 CLMU80 9955864 IC50 = 0.3 nM T61744 CV6TO1 9995407 IC50 = 27.2 nM T61744 CA9YF5 9998837 IC50 = 271 nM T61744 CFPR64 9999276 EC50 = 20 nM T61744 C53HZC 9999401 IC50 = 587 nM T61744 C3A6RV 10027487 IC50 = 0.57 nM T61744 C3VT5F 10065530 IC50 = 25 nM T61744 C8T3LV 10090103 IC50 = 537 nM T61744 C6T4JS 10091127 IC50 = 587 nM T61744 CBUX03 10113183 IC50 = 0.34 nM T61744 CFY9M8 10115569 IC50 = 0.62 nM T61744 CK5C9Z 10119563 IC50 = 0.8 nM T61744 C1EVS3 10119564 IC50 = 1 nM T61744 C83BSD 10128917 IC50 = 0.2 nM T61744 CWDR26 10129145 IC50 = 1.6 nM T61744 CME68G 10152836 IC50 = 0.1 nM T61744 C0PVT2 10153372 IC50 = 2.1 nM T61744 C7D5IT 10158829 IC50 = 107 nM T61744 CB6V1X 10162604 IC50 = 0.5 nM T61744 C75JIV 10167216 IC50 = 0.8 nM T61744 CBT4P1 10177031 IC50 = 35 nM T61744 C3X9DK 10183196 IC50 = 11.8 nM T61744 CUXV40 10183769 IC50 = 0.3 nM T61744 CY9HS7 10185841 IC50 = 0.16 nM T61744 CVUZ36 10195164 IC50 = 5.6 nM T61744 C8LYH6 10196396 IC50 = 0.3 nM T61744 CSQ16M 10196596 IC50 = 1 nM T61744 CTV6F9 10196609 IC50 = 0.3 nM T61744 CTZ7Q8 10196916 IC50 = 0.6 nM T61744 CZG54F 10197046 IC50 = 15 nM T61744 CE5LH4 10199681 IC50 = 27 nM T61744 C61CZK 10205978 IC50 = 52 nM T61744 CPU09I 10210579 IC50 = 0.9 nM T61744 CX9LV3 10232106 IC50 = 4.8 nM T61744 CI5Y3F 10254618 IC50 = 0.88 nM T61744 C7RH4B 10270013 IC50 = 242 nM T61744 CGRQ23 10274114 IC50 = 1.54 nM T61744 CHY71P 10274246 IC50 = 0.75 nM T61744 C48ENU 10289786 IC50 = 10 nM T61744 CT5FL2 10289848 IC50 = 0.1 nM T61744 C90DYG 10297996 IC50 = 6.2 nM T61744 CECW14 10301548 IC50 = 0.2 nM T61744 C5IF9A 10312566 IC50 = 1.5 nM T61744 CB71WD 10322207 IC50 = 30 nM T61744 CJ7YZ9 10345293 IC50 = 0.32 nM T61744 C5OQ3Z 10407016 IC50 = 148 nM T61744 C9A1JH 10432102 IC50 = 371 nM T61744 C23HSK 10451184 IC50 = 59 nM T61744 CD09NL 10451631 IC50 = 364 nM T61744 CV6FS0 10456505 IC50 = 0.4 nM T61744 C2GM8H 10531401 IC50 = 250 nM T61744 C1RG7I 10545177 IC50 = 3800 nM T61744 C7G1BH 10547592 IC50 > 10000 nM T61744 CZ15HV 10571743 IC50 = 770 nM T61744 C8RN0L 10611778 IC50 > 10000 nM T61744 CJQZ06 10646520 IC50 = 15 nM T61744 CHU62M 10661230 IC50 = 279 nM T61744 CRJ79L 10664015 IC50 = 120 nM T61744 CO4AP8 10682163 IC50 > 10000 nM T61744 CF2BR1 10691724 IC50 = 1400 nM T61744 CNB35R 10805427 IC50 = 9500 nM T61744 CDL73U 10810934 IC50 = 1800 nM T61744 CFT6Y4 10837787 IC50 = 3.3 nM T61744 C3DMA0 10841260 IC50 = 35 nM T61744 C9QUV7 10863652 IC50 = 1 nM T61744 C0A7DI 11017241 IC50 = 48 nM T61744 C5P8RW 11048955 IC50 = 1.6 nM T61744 CLF67W 11268574 IC50 = 730 nM T61744 C45VZC 11438405 IC50 > 16000 nM T61744 CXO38Q 11493078 IC50 = 21000 nM T61744 CQ8G9F 11525525 IC50 = 5.4 nM T61744 CS5U1Z 11532316 IC50 = 20 nM T61744 C6UMB2 11532832 IC50 = 43 nM T61744 C3G1BO 11604203 IC50 = 2560 nM T61744 CE24AU 11626787 IC50 = 97 nM T61744 C0BD7Q 11628421 IC50 = 5 nM T61744 C37TWP 11633996 IC50 = 4.5 nM T61744 COLF16 11639342 IC50 = 2900 nM T61744 C8U5VK 11641556 IC50 = 74 nM T61744 C8EX6Z 11648288 IC50 = 19 nM T61744 C83NLR 11648915 IC50 = 18 nM T61744 CX2ZD7 11650267 Ki > 1000 nM T61744 CFM64H 11662453 IC50 = 6.7 nM T61744 CR8CQ7 11669507 IC50 = 2330 nM T61744 CQPW60 11705339 IC50 = 9 nM T61744 C0I5BW 11711290 IC50 = 97 nM T61744 CVJ10R 11713455 IC50 = 23 nM T61744 CP7EV6 11731453 IC50 = 0.4 nM T61744 CROY49 11754228 IC50 = 0.54 nM T61744 CC92YE 11755033 IC50 = 0.53 nM T61744 CUK49V 11988837 Ki = 240 nM T61744 CFIO49 11988967 Ki = 1300 nM T61744 CS4XN7 11988968 Ki = 9900 nM T61744 CAEF17 11988969 Ki = 3400 nM T61744 C2IY1E 11988971 Ki = 1500 nM T61744 C2D0NG 11989101 Ki = 930 nM T61744 C65ABT 11989102 Ki = 1200 nM T61744 CT2SJ1 11989104 Ki = 65 nM T61744 C1B4XD 11992634 IC50 > 2000 nM T61744 CPX16N 11993169 IC50 > 2000 nM T61744 C7BE0Q 12991318 IC50 = 9.2 nM T61744 C7QY9B 13747863 IC50 = 160 nM T61744 C40KZA 15434926 IC50 = 250 nM T61744 C4ESY5 15942639 IC50 = 0.5 nM T61744 C6VN5F 16067799 IC50 = 20 nM T61744 CMB3Z5 16067906 IC50 = 0.3 nM T61744 C31LJY 16103072 IC50 = 770 nM T61744 CXFT59 17757146 IC50 = 6.7 nM T61744 CBX29P 17989733 IC50 = 160 nM T61744 C1PZ8C 18734933 IC50 = 107 nM T61744 C8MPD3 19361675 IC50 = 590 nM T61744 CD91IV 19959342 IC50 = 40 nM T61744 CI5Y7D 19959346 IC50 = 47 nM T61744 CI70YS 19959348 IC50 = 172 nM T61744 C3L0DW 19959377 IC50 = 40 nM T61744 CG2VE4 19959383 IC50 = 17 nM T61744 CH10ZO 19959396 IC50 = 389 nM T61744 C7RXF4 20583506 IC50 = 65 nM T61744 CT68OG 20640412 IC50 = 0.3 nM T61744 C61MGH 20640414 IC50 = 0.6 nM T61744 C9DE6Y 20814950 IC50 = 3.4 nM T61744 CCD06M 21198161 IC50 = 70000 nM T61744 C1UL4Q 21251043 IC50 = 2.3 nM T61744 C4MPA2 21251047 IC50 = 0.8 nM T61744 CVX96E 21251056 IC50 = 31 nM T61744 CK14OA 21251062 IC50 = 1.2 nM T61744 C62PHJ 21251066 IC50 = 5.8 nM T61744 C82MXB 21251069 IC50 = 18 nM T61744 CW7X0P 21251089 IC50 = 9.3 nM T61744 CUT04Q 21251090 IC50 = 1.2 nM T61744 C3M5NF 21865580 IC50 = 3.1 nM T61744 C4CWR6 21865595 IC50 = 15 nM T61744 C6T5NZ 21865599 IC50 = 1.8 nM T61744 CULE52 21865620 IC50 = 0.6 nM T61744 CINH54 21865627 IC50 = 3.5 nM T61744 CMHF08 22083604 IC50 = 1.7 nM T61744 C34FLM 22083724 IC50 = 0.47 nM T61744 CWIT18 22083784 IC50 = 0.3 nM T61744 CR4T9J 22337182 Ki > 1000 nM T61744 CMZH62 22391985 IC50 = 141 nM T61744 CBD0R8 22391998 IC50 > 1000 nM T61744 CD48PX 23218492 IC50 = 50.7 nM T61744 CW96SI 23624262 IC50 > 1000 nM T61744 C9WGI4 24802717 IC50 = 5000 nM T61744 C6EQG2 24963293 IC50 > 2000 nM T61744 C4J0YD 25196719 IC50 = 7830 nM T61744 CICF39 42629702 IC50 > 10000 nM T61744 CM3X9S 42629827 IC50 > 1000 nM T61744 CQN26J 42629945 IC50 > 10000 nM T61744 C6O5FX 42630062 IC50 > 10000 nM T61744 C71ZNR 42630180 IC50 = 6350 nM T61744 C4RHY0 42630191 IC50 > 10000 nM T61744 CT6RS9 42630192 IC50 > 5000 nM T61744 CYZL43 42630317 IC50 > 10000 nM T61744 CH42OZ 42630318 IC50 > 10000 nM T61744 C7X5AH 42630437 IC50 = 2650 nM T61744 C46EUM 42639959 Ki = 500 nM T61744 CYZW13 42640117 Ki = 200 nM T61744 CRG8U9 42640266 Ki = 330 nM T61744 COL3R0 42640268 Ki = 460 nM T61744 CK06QZ 42640446 Ki = 420 nM T61744 C5Q0IN 42647289 IC50 = 1.5 nM T61744 CA93LT 44142087 IC50 = 32 nM T61744 CIM96B 44142088 IC50 = 26 nM T61744 CJL04E 44142089 IC50 = 33 nM T61744 CAF2R8 44142090 IC50 = 13 nM T61744 C4D8GB 44142091 IC50 = 35 nM T61744 CSCD90 44142093 IC50 = 21 nM T61744 C39VDQ 44142094 IC50 = 6.1 nM T61744 CL23UQ 44142095 IC50 = 35 nM T61744 C41TSG 44142096 IC50 = 37 nM T61744 CHN08R 44142097 IC50 = 53 nM T61744 C38OYW 44142098 IC50 = 11 nM T61744 CG50DL 44142099 IC50 = 20 nM T61744 CR0D2J 44142100 IC50 = 9.8 nM T61744 C6YR1W 44142101 IC50 = 11 nM T61744 C0V3DP 44142102 IC50 = 7.1 nM T61744 C3SO0L 44142103 IC50 = 3.4 nM T61744 CNIE98 44143458 IC50 = 3 nM T61744 CN2RH8 44143459 IC50 = 7.3 nM T61744 C6MN3V 44143460 IC50 = 11 nM T61744 CQGL19 44143461 IC50 = 3.8 nM T61744 CJ6Q4M 44143462 IC50 = 8.6 nM T61744 CI65DL 44143463 IC50 = 13 nM T61744 CL10UX 44143464 IC50 = 45 nM T61744 CEAU38 44143465 IC50 = 80 nM T61744 C20PNS 44143466 IC50 = 6.7 nM T61744 CW2M7D 44281818 IC50 = 137 nM T61744 C2OR5C 44281838 IC50 = 31 nM T61744 C82QVM 44281839 IC50 = 113 nM T61744 CGU30F 44281858 IC50 = 54.6 nM T61744 C8EKD5 44281860 IC50 = 5 nM T61744 CY45SE 44281877 IC50 = 9 nM T61744 CLCR07 44281889 IC50 = 102 nM T61744 CC2BT4 44281894 IC50 = 2.5 nM T61744 CX5U6W 44281908 IC50 = 12 nM T61744 CFYC79 44281910 IC50 = 5 nM T61744 C8O7RM 44281936 IC50 = 3 nM T61744 C3L6ZM 44281965 Ki = 1170 nM T61744 C29VCQ 44282028 Ki > 8000 nM T61744 CMZN79 44282072 IC50 = 58 nM T61744 C1F0JV 44282073 IC50 = 259 nM T61744 C65WGQ 44282077 IC50 = 5 nM T61744 C5KO0D 44282092 IC50 = 27 nM T61744 CMGV57 44282109 IC50 = 16 nM T61744 CJ4BV9 44282159 IC50 = 8 nM T61744 C4B8OC 44282160 IC50 = 158 nM T61744 CDC8N7 44282176 IC50 = 7.5 nM T61744 C6VU2A 44282235 IC50 = 2.8 nM T61744 C0VF3M 44282255 IC50 = 13 nM T61744 CN8IE2 44282270 IC50 = 110 nM T61744 CXP2K7 44282282 IC50 = 7 nM T61744 CA10HR 44282287 IC50 = 7 nM T61744 CT7F0Y 44282295 IC50 = 11 nM T61744 CEC1N5 44282297 IC50 = 3.1 nM T61744 CKT21Y 44282311 IC50 > 1000 nM T61744 C6K8DH 44282324 IC50 = 10 nM T61744 CMI39O 44282341 IC50 = 24 nM T61744 C8O7AY 44282345 IC50 = 16 nM T61744 C8ES4L 44282358 IC50 = 11 nM T61744 C30XBI 44282368 IC50 = 7.5 nM T61744 C2G7MQ 44282374 IC50 = 9.6 nM T61744 C0SF6D 44282388 IC50 = 4 nM T61744 C5LIE4 44282409 IC50 = 7 nM T61744 CFW60R 44282463 Ki = 423 nM T61744 C63NSP 44282464 IC50 = 8 nM T61744 CHU65T 44282472 IC50 = 4.8 nM T61744 C4TJ5W 44282474 IC50 = 0.8 nM T61744 CDJ71W 44282483 IC50 = 510 nM T61744 C5UF7Z 44282647 IC50 = 2.2 nM T61744 CFKO90 44282699 IC50 = 44 nM T61744 CNQG84 44282705 IC50 = 8.6 nM T61744 CGP95H 44282706 IC50 = 53 nM T61744 CVS3B9 44282707 IC50 = 772 nM T61744 C5DG9T 44282723 IC50 = 410 nM T61744 C1BNZ2 44282725 IC50 = 0.5 nM T61744 CX7U8F 44282737 IC50 = 32 nM T61744 CSC14U 44282738 IC50 = 13 nM T61744 CAG0N4 44282741 IC50 = 19 nM T61744 CPX83U 44282742 IC50 = 22 nM T61744 C8NK2W 44282743 IC50 = 890 nM T61744 CU69NA 44300149 IC50 = 23 nM T61744 CO7BU3 44300524 IC50 = 6 nM T61744 C5TMC6 44300777 IC50 = 3 nM T61744 C6X2QN 44300789 IC50 = 102 nM T61744 C70XSQ 44317802 IC50 = 2.1 nM T61744 C2SLH8 44324331 IC50 = 9.8 nM T61744 C8PNR4 44329482 IC50 > 100000 nM T61744 CUFO76 44329511 IC50 = 540 nM T61744 CA1R5M 44329613 IC50 = 2900 nM T61744 CHR0G3 44329633 IC50 > 100000 nM T61744 CT3M4H 44329639 IC50 = 630 nM T61744 CXUC09 44329640 IC50 = 500 nM T61744 CA5MY8 44329642 IC50 = 1300 nM T61744 CSD45M 44329651 IC50 = 70 nM T61744 CUA7P5 44329666 IC50 = 130 nM T61744 C26ZAE 44329668 IC50 = 3300 nM T61744 C1T7JL 44329669 IC50 = 23500 nM T61744 C2M3QE 44329683 IC50 = 250 nM T61744 C9R0OI 44329684 IC50 = 14000 nM T61744 CWM23U 44329685 IC50 > 10000 nM T61744 CQ2WU3 44329686 IC50 = 85 nM T61744 CMF1J2 44329702 IC50 = 2300 nM T61744 C5YO6L 44329893 IC50 = 5400 nM T61744 CT1C4U 44329894 IC50 = 900 nM T61744 CVM96L 44332873 IC50 = 57 nM T61744 C68HRY 44332874 IC50 = 42 nM T61744 CV1GM2 44332875 IC50 = 38 nM T61744 CXMT40 44332880 IC50 = 2.7 nM T61744 CCM9K0 44332890 IC50 = 27 nM T61744 CKYM84 44332908 IC50 = 18 nM T61744 CIFZ49 44332982 IC50 = 4.4 nM T61744 CU3J2V 44332983 IC50 = 39 nM T61744 CM9ON6 44333328 IC50 = 32 nM T61744 C8YLH3 44339585 IC50 = 370 nM T61744 CST6X1 44339599 IC50 = 120 nM T61744 CND03T 44339619 IC50 = 190 nM T61744 CREM43 44339632 IC50 = 770 nM T61744 C3W8ER 44339633 IC50 = 5000 nM T61744 CA69CV 44339676 IC50 = 740 nM T61744 C1PNH6 44377118 IC50 = 12 nM T61744 CJH19Q 44377130 IC50 = 8.3 nM T61744 CU37PB 44377131 IC50 = 16 nM T61744 C5XT3C 44377148 IC50 = 33 nM T61744 C9IQ7P 44377173 IC50 = 2.3 nM T61744 CWZR92 44377295 IC50 = 1.5 nM T61744 C52QTW 44377340 IC50 = 7.8 nM T61744 CI6M9X 44377348 IC50 = 1.7 nM T61744 C68RAF 44377445 IC50 = 31 nM T61744 CLMW27 44405467 IC50 = 0.5 nM T61744 CR05OY 44405507 IC50 = 1.5 nM T61744 C7OA9V 44405510 IC50 = 0.4 nM T61744 CFY36C 44410864 IC50 = 1.7 nM T61744 CT1JW4 44410870 IC50 = 0.1 nM T61744 C3EI4T 44410882 IC50 = 78 nM T61744 C7NKA2 44410914 IC50 = 16 nM T61744 CSF31I 44562336 IC50 = 0.8 nM T61744 CJD73U 44565305 Ki > 1000 nM T61744 CL62PK 44588589 IC50 = 0.45 nM T61744 CMI7N1 44588590 IC50 = 0.06 nM T61744 CP9QH1 44588591 IC50 = 15.3 nM T61744 CLZ05M 44588592 IC50 = 0.17 nM T61744 C09TKD 44589077 IC50 = 3.54 nM T61744 CW14SN 44589078 IC50 = 66.5 nM T61744 C6XZH8 44589079 IC50 > 1000 nM T61744 CJ3Y9G 46238781 Ki = 37000 nM T61744 CBT91W 46240282 Ki = 18000 nM T61744 CF0PI3 46915888 IC50 = 6.4 nM T61744 C3P2IN 46933992 IC50 = 63.7 nM T61744 CB2HS9 46933993 IC50 = 5.7 nM T61744 CZ7C3F 46933994 IC50 = 12.8 nM T61744 CQ5NF4 49780548 IC50 = 18 nM T61744 C9H4BC 49780549 IC50 = 67 nM T61744 CHA5Z0 49821469 IC50 > 1000 nM T61744 C1AYP0 49821627 IC50 > 500 nM T61744 C85AXR 49821714 IC50 > 1000 nM T61744 C0EH7V 49865602 IC50 = 307 nM T61744 C89UPD 49865603 IC50 = 350 nM T61744 CV81PG 49865604 IC50 = 224 nM T61744 C43XGJ 49865605 IC50 = 166 nM T61744 CIT05Z 49865642 IC50 = 819 nM T61744 C5OI1V 49865643 IC50 = 60.4 nM T61744 C19JZB 49866243 IC50 = 9.9 nM T61744 CU5B8G 49866268 IC50 = 4.6 nM T61744 CSYL46 49866269 IC50 = 126 nM T61744 CI3F7K 49866270 IC50 = 319 nM T61744 C7V8DY 49866271 IC50 = 338 nM T61744 CCJ7I1 49866272 IC50 = 122 nM T61744 CVIJ94 52997854 Ki = 69000 nM T61744 CAWD97 53237026 IC50 = 5400 nM T61744 CC80RP 53237027 IC50 = 24000 nM T61744 C6ZQC8 53237028 IC50 = 12000 nM T61744 C8Z9VY 53237241 EC50 = 500 nM T61744 CFS95I 53237242 IC50 = 2400 nM T61744 CB0ET1 53237243 EC50 = 2100 nM T61744 CS3E0K 53237455 IC50 = 38000 nM T61744 C41ATC 53237456 IC50 = 44000 nM T61744 C6UR2P 53237457 EC50 = 5600 nM T61744 C4NJS7 53237458 IC50 = 6400 nM T61744 CW5QR9 53237459 EC50 = 4600 nM T61744 C67ETO 53237460 IC50 = 8200 nM T61744 CQF4R9 54760727 Ki = 250 nM T61744 C3GL0H 54760728 Ki = 220 nM T61744 CHT86A 56642417 IC50 = 16.3 nM T61744 CBV60W 56642529 IC50 = 4.8 nM T61744 CKGD94 56642530 IC50 = 36 nM T61744 CKTD52 56642531 IC50 = 5 nM T61744 C4G6TL 56642532 IC50 = 28 nM T61744 CRK35Q 56642533 IC50 = 5 nM T61744 CF7P1Y 56642534 IC50 = 62 nM T61744 CP9CD7 56642658 IC50 = 22 nM T61744 CM8U9E 56642659 IC50 = 6.2 nM T61744 CAN50G 56642660 IC50 = 0.9 nM T61744 C4TGL7 56648496 IC50 > 1000 nM T61744 CH6C3L 56648679 IC50 > 10000 nM T61744 CCY79V 56648680 IC50 = 2590 nM T61744 CNE96P 56648857 IC50 > 10000 nM T61744 CX86AQ 56648859 IC50 > 5000 nM T61744 C1AND4 56659469 IC50 = 17 nM T61744 CGWH19 56662928 IC50 = 32 nM T61744 CQT17K 56662929 IC50 = 0.51 nM T61744 CLMG01 56662930 IC50 = 0.52 nM T61744 CL1U3W 56666405 IC50 = 0.66 nM T61744 C5H9XA 56669821 IC50 = 0.55 nM T61744 CIX9M0 56673307 IC50 = 0.46 nM T61744 CTY48D 56673902 IC50 = 4.6 nM T61744 CEO42M 56676640 IC50 = 0.58 nM T61744 C2CRW3 56679969 IC50 = 1 nM T61744 CT8A6K 56683302 IC50 = 0.35 nM T61744 C0YD3P 56928304 IC50 > 5000 nM T61744 C8RO6A 56929788 IC50 > 1000 nM T61744 C2ZD7G 57390975 IC50 = 471 nM T61744 CHB1V2 57390976 IC50 = 994 nM T61744 CO75IQ 57390977 IC50 = 477 nM T61744 C6EI3A 57390978 IC50 = 362 nM T61744 C5CLS9 57390979 IC50 > 1000 nM T61744 C61WPI 57390980 IC50 > 1000 nM T61744 CDHJ84 57390991 IC50 > 1000 nM T61744 C6W8KX 57390992 IC50 > 1000 nM T61744 CES36G 57390993 IC50 > 1000 nM T61744 C01JFV 57390994 IC50 > 1000 nM T61744 CODM26 57390995 IC50 > 1000 nM T61744 CD52CA 57391118 IC50 > 2000 nM T61744 C68NJH 57392756 IC50 > 5000 nM T61744 CJPE69 57392757 IC50 = 560 nM T61744 CN85ZR 57392758 IC50 > 1000 nM T61744 C2A5RM 57392759 IC50 = 458 nM T61744 C0F7ON 57392760 IC50 = 481 nM T61744 CLV6C2 57392761 IC50 > 1000 nM T61744 C5IAB9 57392762 IC50 > 1000 nM T61744 CI9K4B 57392763 IC50 > 1000 nM T61744 CT67RF 57392774 IC50 > 1000 nM T61744 CPNH58 57392775 IC50 > 1000 nM T61744 CJV0C8 57392776 IC50 = 362 nM T61744 C89ZVD 57392777 IC50 = 156 nM T61744 C0LZ1P 57392778 IC50 = 1420 nM T61744 CD3QS0 57394488 IC50 = 379 nM T61744 C8DIO6 57394489 IC50 > 1000 nM T61744 CPA7C8 57394490 IC50 > 1000 nM T61744 C52PKN 57394491 IC50 = 430 nM T61744 C0G9QL 57394492 IC50 = 1060 nM T61744 CNS3R5 57394502 IC50 > 1000 nM T61744 C8HNQ3 57394503 IC50 > 1000 nM T61744 C85UHM 57394504 IC50 > 1000 nM T61744 C7SX3Y 57394505 IC50 > 1000 nM T61744 CHE68W 57394506 IC50 > 1000 nM T61744 C1V0IE 57394507 IC50 = 580 nM T61744 C0F6OX 57394508 IC50 = 73 nM T61744 CJ6E9Q 57396249 IC50 = 1520 nM T61744 CI8S6J 57396252 IC50 = 516 nM T61744 CZ3V0H 57396253 IC50 = 274 nM T61744 CT9XE7 57398056 IC50 > 1000 nM T61744 COQJ51 57398057 IC50 = 90 nM T61744 CFB2P9 57399706 IC50 = 442 nM T61744 C2B1AF 57399707 IC50 > 1000 nM T61744 C7MWD1 57399708 IC50 = 201 nM T61744 C8UZ1R 57399715 IC50 > 1000 nM T61744 CO3AG1 57399716 IC50 = 161 nM T61744 CX27HZ 57401470 IC50 > 1000 nM T61744 C8QU1A 57401471 IC50 = 568 nM T61744 C0FW5U 57401478 IC50 = 402 nM T61744 C1WS7F 57403204 IC50 = 506 nM T61744 C0KL7Y 57403205 IC50 = 1330 nM T61744 C2UX3A 57403206 IC50 = 219 nM T61744 CP0L9U 57403207 IC50 > 1000 nM T61744 CX4M5I 57403214 IC50 > 1000 nM T61744 COYT07 57403215 IC50 > 5000 nM T61744 C0C6TW 57403216 IC50 > 1000 nM T61744 C3D1OC 57403217 IC50 = 3560 nM T61744 CCA5S3 57403218 IC50 > 1000 nM T61744 C6DA0M 57403219 IC50 > 1000 nM T61744 CJ6TS1 57403220 IC50 = 979 nM T61744 CB4PT8 57403221 IC50 = 385 nM T61744 C2MA7Z 58456655 Ki = 930 nM T61744 CW24YS 59190451 IC50 < 10 nM T61744 CEI8A5 59190544 IC50 < 10 nM T61744 C9GA7N 59548042 Ki = 4100 nM T61744 C4ZEH9 68578314 IC50 = 3370 nM T61744 CEI21Q 70319863 Ki = 44000 nM T61744 C9GR3L 71153436 IC50 > 10000 nM T61744 CJ62MK 71451776 IC50 = 64 nM T61744 C2UK6B 71451779 IC50 = 159 nM T61744 CE1TP4 71460359 EC50 = 270 nM T61744 CJ3Z7K 71460703 IC50 = 2.1 nM T61744 C4GNJ3 71598545 IC50 = 0.81 nM T61744 CKIH79 71727293 IC50 = 156 nM T61744 CC90DN 71727294 IC50 = 104 nM T61744 CSV3F4 71727397 IC50 = 87 nM T61744 CSR5Z9 71727398 IC50 = 40 nM T61744 CIQ3D0 71727399 IC50 = 54 nM T61744 C01ANQ 71727400 IC50 = 44 nM T61744 CKXA98 71727401 IC50 = 60 nM T61744 C2K4DO 71727402 IC50 = 149 nM T61744 C6I0CF 71727403 IC50 = 1040 nM T61744 CW32VD 71727499 IC50 = 165 nM T61744 CT5XM7 71727500 IC50 = 126 nM T61744 C48TIQ 71727501 IC50 = 668 nM T61744 C3J8XI 71727502 IC50 = 563 nM T61744 CZ3X1I 71727503 IC50 = 19 nM T61744 CO94RY 71727504 IC50 = 38 nM T61744 C4X1MC 71727505 IC50 = 19 nM T61744 C85ODL 71727506 IC50 = 4.4 nM T61744 CQ93BY 71727507 IC50 > 1000 nM T61744 CD1IX9 71727608 IC50 = 232 nM T61744 CDE7W9 71727609 IC50 = 153 nM T61744 CLU28C 71727610 IC50 = 59 nM T61744 C2I7RY 71727611 IC50 = 56 nM T61744 CT6CN3 71727612 IC50 = 18 nM T61744 C62UOR 71727613 IC50 = 38 nM T61744 C42SID 71727614 IC50 = 6.6 nM T61744 CQ3JC7 71727615 IC50 = 12 nM T61744 C15JYG 71727720 IC50 = 1.7 nM T61744 C7BTQ8 71727721 IC50 = 1 nM T61744 CC8SE6 71727722 IC50 = 4.9 nM T61744 C61YGS 71727723 IC50 = 1.4 nM T61744 C1WQ4J 71727724 IC50 = 0.42 nM T61744 CGBO18 71727725 IC50 = 0.15 nM T61744 CDAG28 71727726 IC50 = 0.2 nM T61744 C7QAM0 71727727 IC50 = 1.6 nM T61744 CS3BJ5 71727841 IC50 = 3.6 nM T61744 C4XMW9 71727842 IC50 = 6.5 nM T61744 CS4V7T 71727843 IC50 = 1.1 nM T61744 CVJ3T0 71727844 IC50 = 2.4 nM T61744 CIBX67 71727845 IC50 = 0.89 nM T61744 C52ZYE 71727846 IC50 = 2.7 nM T61744 CQ3GD7 72704434 Ki = 160 nM T61744 CRJ8D4 90665374 IC50 = 3850 nM T61744 C4RN9B 90667924 EC50 = 11660 nM T61744 CG5HV8 90668361 IC50 = 199000 nM T61744 C2HQ7I 90668362 IC50 = 4180 nM T61744 CDB74T 90668364 IC50 = 5600 nM T61744 C5TL8H 118725359 IC50 = 25400 nM T61744 CE49ML 118725368 IC50 = 40300 nM T61744 C0I8FH 118875015 Ki = 1200 nM T61744 CJKO62 122193703 IC50 = 8350 nM T61744 C9W1JO 122193704 IC50 = 4090 nM T61744 C2MNX0 122193705 IC50 = 460 nM T61744 C5EHB7 122193706 IC50 = 1010 nM T61744 C5WI6U 122193707 IC50 = 2220 nM T61744 COT0R6 122193708 IC50 = 1440 nM T61744 CJF36H 122193709 IC50 = 1570 nM T61744 C0J6MS 122193710 IC50 = 9890 nM T61744 C0XLR7 122193711 IC50 = 5970 nM T61744 CC9I0U 122193712 IC50 = 1570 nM T61744 CX30HD 122193713 IC50 = 1760 nM T61744 C6IJH8 122193928 IC50 = 3720 nM T61744 CNT17O 122193929 IC50 = 4770 nM T61744 C6Q5UO 122193930 IC50 = 12300 nM T61744 C1SWM0 122193931 IC50 = 8360 nM T61744 C9JSX0 122193932 IC50 = 15000 nM T61744 C6GI3B 122193933 IC50 = 12400 nM T61744 C9PTW4 122193934 IC50 = 1860 nM T61744 C5FKM8 122193935 IC50 = 9730 nM T61744 C6B5XA 124655957 Ki = 8400 nM T61744 C6WS7G 127025427 Ki = 860 nM T61744 C2WBK3 127025428 Ki = 18000 nM T61744 CLR0X4 127025703 Ki = 700 nM T61744 C1OIN6 127026000 Ki = 3000 nM T61744 CV9MQ0 127026292 Ki = 12000 nM T61744 COK0Y4 127026293 Ki = 13000 nM T61744 CNZ94R 127026294 Ki > 100000 nM T61744 CJS3H9 127026295 Ki = 30000 nM T61744 CP2N0X 127026298 Ki = 9800 nM T61744 CT98XU 127026299 Ki = 2000 nM T61744 CU5Y8A 127026300 Ki = 8400 nM T61744 C9V6TE 127026301 Ki = 390 nM T61744 CY6N3Q 127026600 Ki > 100000 nM T61744 C1ZPB2 127026608 Ki = 4100 nM T61744 CYD1I3 127026875 Ki = 5500 nM T61744 CWX74A 127026876 Ki = 6300 nM T61744 CU73HG 127027157 Ki = 2400 nM T61744 CX8JA4 127027158 Ki = 4300 nM T61744 CLK93H 127027159 Ki = 1100 nM T61744 C62JMC 127027160 Ki = 6200 nM T61744 CDSU28 127027161 Ki = 2600 nM T61744 CPE30I 127027162 Ki = 5500 nM T61744 CM0W5L 127027163 Ki = 1600 nM T61744 CQZ28R 127027169 Ki = 4600 nM T61744 C0FO7D 127027178 Ki = 8400 nM T61744 CJ40XR 127027474 Ki = 370 nM T61744 CE1BS3 127027475 Ki = 4000 nM T61744 CQS23D 127027476 Ki = 740 nM T61744 CQ49HJ 127027485 Ki = 770 nM T61744 CV85XN 127027487 Ki = 780 nM T61744 C5OW1G 127028159 Ki = 1200 nM T61744 C8P7IE 127028160 Ki = 3100 nM T61744 CTE87U 127028161 Ki > 100000 nM T61744 C3BZ7F 127028162 Ki = 4700 nM T61744 C4UR7D 127038167 IC50 > 1000 nM T61744 C4H2TJ 127038168 IC50 > 1000 nM T61744 CL9JT8 127038169 IC50 > 1000 nM T61744 CJPX60 127038509 IC50 = 1000 nM T61744 C26EAG 127038511 IC50 > 841 nM T61744 CTM9E4 127038512 IC50 > 1000 nM T61744 C6AQ2U 127038513 IC50 > 1000 nM T61744 CV1FM0 127038868 IC50 > 1000 nM T61744 CADU23 127038869 IC50 < 1000 nM T61744 CW2HR1 130366728 IC50 = 2 nM T61744 C2ALN7 130366739 IC50 = 31.9 nM T61744 CQJN83 130366758 IC50 = 241 nM T61744 CDAF16 130380472 IC50 = 115 nM T61744 C18KLO 130380505 IC50 = 188 nM T61744 C5XCO1 130380512 IC50 = 12 nM T61744 CT2E8Q 130380575 IC50 = 20.6 nM T61744 C2P1IU 134129996 IC50 = 95 nM T61744 CLE03O 134130328 IC50 = 117 nM T61744 CSN6J0 134130563 IC50 = 76 nM T61744 C0A1CZ 134131162 IC50 = 126 nM T61744 C3R8SE 135457869 IC50 > 10000 nM T61744 C1RK8U 135815296 Ki = 179 nM T61744 CTX54Z 135896326 IC50 > 10000 nM T61744 CNX76Q 135927702 Ki = 18000 nM T61744 CIW37T 136035260 IC50 = 3300 nM T61744 C12UMG 136059728 IC50 > 1000 nM T61744 C2VO1H 136132220 Ki = 147 nM T61744 C8PG9Q 136132221 Ki = 137 nM T61744 CUI4W9 136132222 Ki = 103 nM T61744 CST26Q 136132223 Ki = 208 nM T61744 CQ27TM 136132224 Ki = 15200 nM T61744 CMIY85 136132225 Ki = 155 nM T61744 C7J3IT 136132226 Ki = 405 nM T61744 CT3IC8 136132227 Ki = 5200 nM T61744 CYM29K 136132228 Ki = 175 nM T61744 CEM5N1 136132229 Ki > 50000 nM T61744 C4V5AD 136132230 Ki = 225 nM T61744 CJC0X9 136132231 Ki = 3390 nM T61744 COA9T2 136132232 Ki = 113 nM T61744 CQ50CG 136132233 Ki = 309 nM T61744 CY50JV 136132234 Ki = 206 nM T61744 C28IYL 136132235 Ki = 244 nM T61744 CHW75A 136132236 Ki = 166 nM T61744 C9GA2W 136132237 Ki = 1190 nM T61744 C39MDZ 136132238 Ki = 175 nM T61744 CW3FM6 136132239 Ki = 126 nM T61744 C5XBZ6 136132240 Ki = 236 nM T61744 CU8RC1 136132241 Ki = 415 nM T61744 C5NVZ9 136132242 Ki = 271 nM T61744 CF31SZ 136132243 Ki = 223 nM T61744 C21FVA 136180322 IC50 = 3700 nM T61744 CH3DA8 137226424 Ki = 550 nM T61744 CLN2U7 137652270 IC50 = 9900 nM T61744 CSOF52 141737655 IC50 > 10000 nM T61744 C7SRA2 141737657 IC50 > 10000 nM T61744 CMIY07 141737666 IC50 > 10000 nM T61744 CC61SD 141737667 IC50 > 10000 nM T61744 C14CZJ 141737668 IC50 > 10000 nM T61744 CTNG49 141737674 IC50 > 10000 nM T61744 CJ38IC 141737676 IC50 > 10000 nM T61744 C1MC5Z 141737681 IC50 > 10000 nM T61744 CTUL23 141737690 IC50 > 10000 nM T61744 CMW20N 141737696 IC50 > 10000 nM T61744 CO1C4S 141737703 IC50 > 10000 nM T61744 CX9N1P 141737704 IC50 > 10000 nM T61744 C8HEG7 141737705 IC50 > 10000 nM T61744 C1S7HV 142592633 IC50 = 100 nM T61744 CN3OC2 142592634 IC50 = 152 nM T61744 CY64NR 142592636 IC50 = 89 nM T61744 C83XNL 142592649 IC50 = 45 nM T61744 C7XZB1 142592652 IC50 = 284 nM T61744 C9SH7Y 145949856 IC50 = 11800 nM T61744 D01CAY 16038022 IC50 = 560 nM T61744 D01RUN 448055 IC50 = 162 nM T61744 D02FZD 158758 EC50 = 3400 nM T61744 D02NKD 10711281 IC50 = 350 nM T61744 D04XRV 10547238 IC50 = 28 nM T61744 D0J4AT 10990391 IC50 = 2300 nM T61744 D0JD4C 9853498 IC50 = 1.4 nM T61744 D0K4HG 9819356 IC50 = 0.07 nM T61744 D0L0NY 10565073 IC50 = 9 nM T61744 D0N2KP 44339586 IC50 = 44 nM T61744 D0P2HX 9842556 EC50 = 17 nM T61744 D0P2TS 9818682 IC50 = 1800 nM T61744 D0V1IM 9808191 IC50 = 4.2 nM T61744 D0V4WB 149790 IC50 > 16000 nM T61744 D0V8DB 10642995 IC50 = 2.7 nM T61744 D0W7BI 44339577 IC50 = 340 nM T61744 D0W7WV 11039077 IC50 = 0.4 nM T61744 D0Z5SB 10404815 IC50 = 0.2 nM T03691 D09JUG 60490 IC50 = 850 nM T03691 D0E3SH 6918837 IC50 > 10000 nM T03691 D0E7PQ 5311 IC50 = 1670 nM T03691 D0I0EG 44093 IC50 = 3600 nM T03691 D0RA5Q 72172 Ki = 320 nM T03691 D00FHR 9865515 IC50 > 10000 nM T03691 D01UXJ 11609955 IC50 > 10000 nM T03691 D05KED 53340666 IC50 > 10000 nM T03691 D09XIZ 11538455 IC50 > 10000 nM T03691 D0GE5B 56654642 IC50 > 10000 nM T03691 D0GH3Q 9804992 IC50 > 10000 nM T03691 D0L2UQ 49855250 IC50 > 10000 nM T03691 D0M8FD 4261 IC50 > 10000 nM T03691 D0U3EP 445154 IC50 = 366000 nM T03691 D0V0SL 11749858 IC50 > 10000 nM T03691 D0XT6W 6918638 IC50 > 10000 nM T03691 D0Z4RC 24756910 IC50 > 10000 nM T03691 D0J8OC 5186 IC50 = 4400 nM T03691 D05MCS 44473151 IC50 > 100000 nM T03691 D0C0JT 4495 IC50 > 100000 nM T03691 D0X9PW 108092 IC50 = 160 nM T03691 CNG85F 3473 IC50 = 56120 nM T03691 C8HA6K 3994 IC50 = 300 nM T03691 C9D4IO 67861 IC50 > 1000000 nM T03691 C5D8BC 87110 IC50 > 1000000 nM T03691 CM2CV8 97908 IC50 = 17300 nM T03691 CCE6Q7 127419 IC50 = 230 nM T03691 CAE8W7 164472 IC50 = 26 nM T03691 C1UJD0 222746 IC50 = 6 nM T03691 CM94DZ 237561 IC50 > 100000 nM T03691 C9RFL4 244154 IC50 > 100000 nM T03691 C65MQC 461252 Ki = 14000 nM T03691 C6EFN7 803072 IC50 = 1800 nM T03691 CEX3O2 803120 IC50 = 30 nM T03691 C78YTV 934481 IC50 = 2000 nM T03691 C1E5DH 2762293 IC50 > 1000000 nM T03691 CLNU65 2828785 IC50 = 13000 nM T03691 C93LZS 2993547 IC50 = 1650 nM T03691 CDY02V 2994178 IC50 = 120 nM T03691 CZ02EN 3768902 Ki = 360 nM T03691 CD03QL 4566654 IC50 > 18000 nM T03691 C1QWR2 5275725 IC50 > 100000 nM T03691 C47ALD 5275726 IC50 = 15240 nM T03691 CZM7D8 5281794 IC50 = 12540 nM T03691 CH9PD2 5317596 IC50 > 100000 nM T03691 CP1FJ5 6603747 IC50 ~ 20000 nM T03691 CN9UD4 8027171 IC50 > 2000000 nM T03691 CK2Q6E 9804586 IC50 = 75 nM T03691 C86NWC 9820434 IC50 = 2.5 nM T03691 CO7S5D 9822092 IC50 = 27 nM T03691 CP36AE 9838405 Ki = 18 nM T03691 CG9I0Z 9839929 IC50 = 8700 nM T03691 C1TEG2 9862473 IC50 = 2 nM T03691 C1UN7R 9863103 IC50 = 250 nM T03691 C6WI4J 9884772 IC50 = 43 nM T03691 CX28YL 9905882 IC50 = 130 nM T03691 CCB45G 9907252 IC50 = 1800 nM T03691 CK41VD 9909196 IC50 = 1.3 nM T03691 C7DUW1 9909236 IC50 = 0.5 nM T03691 CG4U7A 9927621 IC50 = 4.7 nM T03691 CL42DF 9928236 IC50 = 160 nM T03691 C9UQI6 9949943 IC50 = 2100 nM T03691 C1I3YR 9950170 IC50 = 16 nM T03691 CJ02HL 9975300 IC50 = 590 nM T03691 CF6N4G 9992381 Ki = 15000 nM T03691 CQO56T 9993978 IC50 = 780 nM T03691 CD6Y1N 10041390 IC50 = 20000 nM T03691 CX35YD 10060458 IC50 > 1000000 nM T03691 CGSQ79 10064161 IC50 = 600 nM T03691 C1APE5 10068061 IC50 = 3000 nM T03691 CB98TR 10082805 IC50 = 20000 nM T03691 CR12HX 10084376 IC50 > 5000000 nM T03691 CALN39 10104462 IC50 = 80000 nM T03691 CQI5E0 10249742 Ki = 46 nM T03691 CD50YN 10264885 IC50 = 80000 nM T03691 C84ENL 10331928 IC50 = 140000 nM T03691 CSHT82 10333202 IC50 = 200 nM T03691 C27IBJ 10335303 IC50 = 500 nM T03691 CPI56A 10335638 IC50 = 70 nM T03691 CBVO15 10338219 IC50 = 31 nM T03691 CD4OL8 10357905 IC50 = 3 nM T03691 C1W7XS 10403990 IC50 > 100000 nM T03691 CT6ZV3 10408145 IC50 = 800 nM T03691 CMF79L 10425734 IC50 = 140 nM T03691 C8PWU5 10447524 IC50 = 5 nM T03691 CG7A3I 10492795 IC50 = 260 nM T03691 C68PXT 10495421 IC50 = 9700 nM T03691 CS5GZ6 10517981 IC50 = 700 nM T03691 C23CIJ 10518129 IC50 = 1800 nM T03691 CPA79F 10519454 IC50 = 80 nM T03691 CFX27V 10540733 IC50 > 3000 nM T03691 CF3CE7 10541927 IC50 = 220 nM T03691 CDW5Y2 10542930 IC50 = 37 nM T03691 CC0WG7 10543074 IC50 > 100000 nM T03691 CWT2V9 10564654 IC50 = 670 nM T03691 C59IMZ 10566070 IC50 = 53 nM T03691 CY3LO8 10567027 IC50 > 10000 nM T03691 C95IBS 10568376 IC50 = 7500 nM T03691 C67MWH 10588193 IC50 = 47 nM T03691 CZ2BN4 10589458 IC50 = 77 nM T03691 CY5R6X 10612248 IC50 > 3000 nM T03691 CHX54B 10615292 IC50 = 60 nM T03691 C8YEK2 10636646 IC50 = 630 nM T03691 CS3WQ4 10636647 IC50 = 87 nM T03691 CPW41F 10636648 IC50 = 82 nM T03691 C86MBD 10637703 IC50 = 27 nM T03691 C17QIK 10638789 IC50 = 840 nM T03691 CO1S8X 10638790 IC50 = 9000 nM T03691 CH69UI 10661644 IC50 = 420 nM T03691 CZ4BC5 10665216 IC50 = 4000 nM T03691 CJ21XO 10684790 IC50 = 69 nM T03691 CSH4K1 10685308 IC50 = 55 nM T03691 CZ10AY 10686505 IC50 = 140 nM T03691 CS58YH 10689827 IC50 = 140 nM T03691 CL6CB2 10707436 IC50 > 3000 nM T03691 C7T3PW 10708447 IC50 = 33 nM T03691 CMA64B 10708448 IC50 = 36 nM T03691 CIX0S4 10708509 IC50 = 190 nM T03691 C7VH0L 10708721 IC50 = 370 nM T03691 CPWN38 10709151 IC50 = 480 nM T03691 C4ZPE5 10709281 IC50 = 60 nM T03691 CS8P7F 10711066 IC50 = 20 nM T03691 C0GI5E 10730559 IC50 = 8200 nM T03691 CI25MG 10732505 IC50 = 1500 nM T03691 C4T8CZ 10732657 IC50 > 3000 nM T03691 C9G3EJ 10732658 IC50 = 1600 nM T03691 CI6CO0 10732834 IC50 = 170000 nM T03691 CR79SA 10755814 IC50 = 4300 nM T03691 CB8IF1 10780930 IC50 = 900 nM T03691 CFO35Q 10803836 IC50 > 3000 nM T03691 CVN73F 10804675 IC50 > 25000 nM T03691 C8XI2Y 10825997 IC50 = 250 nM T03691 C1PQ3D 10828770 IC50 > 25000 nM T03691 C3B0YQ 10829025 IC50 = 67 nM T03691 CR85GX 10829026 IC50 = 150 nM T03691 CF20VD 10829285 IC50 = 11 nM T03691 C35WOL 10850487 IC50 = 1800 nM T03691 C05RYX 10850852 IC50 = 40 nM T03691 CY9IW3 10851474 IC50 = 620 nM T03691 C2J0PI 10852867 IC50 = 1200 nM T03691 CI60EV 10860416 IC50 = 18 nM T03691 C7V6MB 10871570 IC50 = 450 nM T03691 C4CD3V 10871680 IC50 = 31 nM T03691 C20NAF 10872321 IC50 = 520 nM T03691 CPCO26 10927769 IC50 = 72 nM T03691 C78NDV 10937169 IC50 = 3300 nM T03691 CVS08M 10946934 IC50 = 2500 nM T03691 CC7Z6E 10958396 IC50 = 3000 nM T03691 C0JMF7 10992112 IC50 = 220 nM T03691 CJO97T 11001501 IC50 = 1.3 nM T03691 CMCG27 11002353 IC50 = 14 nM T03691 CO23SP 11013271 IC50 = 450 nM T03691 C1DH4F 11023863 IC50 = 7 nM T03691 C7HS2X 11035648 IC50 = 10700 nM T03691 CP6N7S 11078398 IC50 = 820 nM T03691 C1D7CR 11088726 IC50 = 110 nM T03691 C65NQO 11089570 IC50 = 250 nM T03691 CC0SH3 11089571 IC50 = 110 nM T03691 C8G0RK 11128579 Ki = 50000 nM T03691 C07QHY 11141513 IC50 = 220 nM T03691 C1HK4Y 11152709 IC50 = 240 nM T03691 C7A4PQ 11155062 IC50 = 66 nM T03691 C3CAP9 11189372 IC50 = 13 nM T03691 CYA5K2 11198512 IC50 = 110 nM T03691 CC25EY 11200344 IC50 = 8 nM T03691 CD98NL 11201443 IC50 = 16 nM T03691 C5SOH9 11210422 IC50 = 9 nM T03691 C6JSO4 11210848 IC50 = 14 nM T03691 CB5YH3 11211303 IC50 = 13 nM T03691 C5TAN7 11223519 IC50 = 12 nM T03691 CP8EW3 11245596 IC50 = 11 nM T03691 C6J1HY 11279206 IC50 = 3000 nM T03691 CXL9R8 11291973 IC50 = 28 nM T03691 CY75TS 11303210 IC50 = 31 nM T03691 CVB45M 11315811 IC50 = 10 nM T03691 CP8Y7T 11328449 IC50 = 70 nM T03691 CI7OV1 11359197 IC50 = 84 nM T03691 CG0NR6 11373792 IC50 = 6 nM T03691 C6I0YP 11416924 IC50 = 8 nM T03691 CQ43TD 11472786 IC50 = 7 nM T03691 C8ZA9F 11484587 IC50 = 14 nM T03691 C02ZGN 11725669 IC50 = 0.8 nM T03691 CQW64B 11741633 IC50 = 10000 nM T03691 CGJY03 11759918 IC50 = 560 nM T03691 C35KOU 11771257 IC50 > 100000 nM T03691 C3H2BR 11777264 IC50 > 100000 nM T03691 C76CLK 11810579 IC50 = 4 nM T03691 CTX2Y6 11816616 IC50 > 500000 nM T03691 CO12QC 11823669 IC50 = 19 nM T03691 CXF68D 11824042 IC50 = 2500 nM T03691 C4V0UA 11824423 IC50 = 7 nM T03691 CLJ39H 14186527 IC50 = 250000 nM T03691 CSTI17 14186529 IC50 ~ 250000 nM T03691 CM23TR 14186530 IC50 > 250000 nM T03691 CR93YB 14186556 IC50 > 100000 nM T03691 CTUS78 14330775 IC50 = 22110 nM T03691 CX7Y8T 15011209 IC50 ~ 100000 nM T03691 C40QWD 16220166 IC50 = 180 nM T03691 CRU8L7 16222641 IC50 = 244 nM T03691 C3VA6I 17830966 IC50 = 280 nM T03691 C9NLR1 18678144 IC50 > 3000 nM T03691 CO9D1Q 18678148 IC50 = 47 nM T03691 CQN50W 18678160 IC50 = 11 nM T03691 CR9LE8 18678176 IC50 = 120 nM T03691 C9R0OD 18678179 IC50 = 560 nM T03691 CT8I2A 18678190 IC50 = 4100 nM T03691 C76FJH 18678194 IC50 = 50 nM T03691 C7FZU1 18678203 IC50 = 210 nM T03691 C68VAJ 18678225 IC50 = 16 nM T03691 CO5UN0 18678229 IC50 = 140 nM T03691 CVD0K2 18678234 IC50 = 1100 nM T03691 CC5N7B 18678235 IC50 = 30 nM T03691 CI35UN 18678241 IC50 = 8 nM T03691 C7X2HU 18678246 IC50 = 470 nM T03691 CA3MH0 18678249 IC50 = 20 nM T03691 C1L9QX 18678253 IC50 = 180 nM T03691 C06TVI 18678260 IC50 = 730 nM T03691 CTL49C 18678268 IC50 = 990 nM T03691 CO94AR 18678296 IC50 = 450 nM T03691 C8BD6E 18678308 IC50 = 210 nM T03691 CC27SW 18678310 IC50 = 87 nM T03691 CI5QC8 18678332 IC50 = 81 nM T03691 CEL7Z9 18678337 IC50 = 40 nM T03691 CBK7J6 18678344 IC50 > 3000 nM T03691 CQTN04 18678345 IC50 = 57 nM T03691 CFI59N 22139205 IC50 = 234000 nM T03691 CB7FD9 22690542 IC50 = 150 nM T03691 CUZ10C 22691264 IC50 > 2000 nM T03691 C9DNF0 22691428 IC50 > 2000 nM T03691 CSQ8L5 22859203 IC50 > 3000 nM T03691 CI9WO3 23553327 IC50 = 82 nM T03691 C8K4WT 23553328 IC50 = 36 nM T03691 CT72CK 23553331 IC50 = 100 nM T03691 CET5I0 23553367 IC50 = 390 nM T03691 CT4WD7 23553368 IC50 = 210 nM T03691 C6TDE3 23553369 IC50 = 47 nM T03691 CLE63F 23644581 Ki = 1.6 nM T03691 C4N3WC 23653293 IC50 = 160 nM T03691 CJ1S5T 24894038 IC50 = 7 nM T03691 C4R6BZ 24901452 IC50 > 1000000 nM T03691 CG5PT3 24901580 IC50 = 54 nM T03691 CWV21J 24901581 IC50 = 140 nM T03691 CUT59D 24901583 IC50 = 350 nM T03691 CUW3S6 24901584 IC50 = 13 nM T03691 C3RZK7 24901585 IC50 = 66 nM T03691 C7TC3P 24901586 IC50 = 11 nM T03691 C4YDO0 24901587 IC50 = 29 nM T03691 CENZ09 24901588 IC50 = 35 nM T03691 C8IP6E 24901589 IC50 = 50 nM T03691 CSD0O9 24901590 IC50 = 17 nM T03691 CZEF59 24901591 IC50 = 12 nM T03691 CRNK57 24901592 IC50 = 21 nM T03691 C81RGS 24901593 IC50 = 27 nM T03691 CQ18FN 24901594 IC50 = 87 nM T03691 C4NE9B 24901595 IC50 = 710 nM T03691 C4S2UQ 24901596 IC50 > 2000 nM T03691 CK20DG 24901597 IC50 > 2000 nM T03691 CE2QF8 24901598 IC50 = 10000 nM T03691 CJY7U1 24901599 IC50 = 5800 nM T03691 C59DJW 24901605 IC50 = 39 nM T03691 C9G7TZ 24901606 IC50 = 60 nM T03691 C2M1XN 24901608 IC50 = 25 nM T03691 CH34SN 24901609 IC50 = 11000 nM T03691 CLC10E 24901610 IC50 = 9400 nM T03691 CJK3L6 24901611 IC50 > 18000 nM T03691 C9VEY0 24901613 IC50 = 730 nM T03691 CPZ2A9 24901618 IC50 = 8000 nM T03691 CGFO40 24901622 IC50 = 17 nM T03691 C2Q5MA 24901623 IC50 > 18000 nM T03691 C21OYW 24901624 IC50 > 18000 nM T03691 CH3DI5 24901628 IC50 = 22 nM T03691 CX2JU1 24901631 IC50 = 22 nM T03691 C4JR0W 24901632 IC50 = 17 nM T03691 CO9B0H 24901633 IC50 = 19 nM T03691 CD5WY3 24901634 IC50 = 20 nM T03691 C2L3BV 24901635 IC50 = 22 nM T03691 C5QM7B 24901636 IC50 = 14 nM T03691 C7GP1I 24901638 IC50 = 5600 nM T03691 C34TSC 24901639 IC50 = 130 nM T03691 CW3X2G 24901640 IC50 = 740 nM T03691 C0GW3Z 24901641 IC50 = 350 nM T03691 CQRW18 24901642 IC50 = 390 nM T03691 CFE80D 24901643 IC50 = 85 nM T03691 CTJU08 24975348 IC50 > 1000000 nM T03691 CX29CK 42641156 IC50 = 68.5 nM T03691 CI06LO 42641832 IC50 = 533 nM T03691 CK8HD3 42641837 IC50 = 23 nM T03691 CAB97U 44129622 IC50 = 966000 nM T03691 CAV83N 44129624 IC50 = 80.5 nM T03691 CZ2JE9 44221318 IC50 = 199000 nM T03691 C2O5KZ 44269754 IC50 = 500 nM T03691 CFPT18 44309803 IC50 = 20000 nM T03691 C4ZN9U 44309819 IC50 > 100000 nM T03691 CQ1G2V 44310089 IC50 > 100000 nM T03691 CNE7R3 44310154 IC50 > 250000 nM T03691 CLZA98 44318490 IC50 = 20000 nM T03691 CFK4L2 44318779 IC50 = 300 nM T03691 CAEK91 44318793 IC50 > 3000 nM T03691 C4A0SW 44318799 IC50 = 8 nM T03691 C9I2SR 44318873 IC50 > 10000 nM T03691 C9OD5A 44318885 IC50 = 30 nM T03691 C06WSQ 44318886 IC50 = 12 nM T03691 CS01DY 44318887 IC50 = 10 nM T03691 C43NSE 44319129 IC50 = 1800 nM T03691 CPNG49 44319130 IC50 = 10 nM T03691 C0IX6S 44341959 IC50 = 110 nM T03691 C0YA2N 44342007 IC50 = 450 nM T03691 C4W1DJ 44342457 IC50 = 52 nM T03691 CR5A2P 44376597 IC50 = 410 nM T03691 CJDX78 44479549 IC50 = 3 nM T03691 C7C1HW 44481057 IC50 = 33 nM T03691 C3NI0V 44481584 IC50 = 7 nM T03691 C46OSV 44481854 IC50 = 733 nM T03691 C9U1KA 44481856 IC50 = 3 nM T03691 CCA93X 44481857 IC50 = 6 nM T03691 CEK5L7 44537807 IC50 = 37 nM T03691 CH1OX6 44563649 IC50 = 386000 nM T03691 CU47WJ 44567641 IC50 = 360 nM T03691 CJ8D5K 44567642 IC50 = 28 nM T03691 CT4O2M 44567643 IC50 = 80 nM T03691 CAG45O 44567644 IC50 = 33 nM T03691 C6OJX8 44567646 IC50 = 47 nM T03691 CG63JX 44567647 IC50 = 40 nM T03691 CL92VA 44567648 IC50 = 440 nM T03691 CY2VX9 44567664 IC50 = 4 nM T03691 CIJK96 44567666 IC50 = 230 nM T03691 CGHN62 44567702 IC50 = 6 nM T03691 C9P1XE 44567703 IC50 = 230 nM T03691 CP4R8L 44567704 IC50 = 70 nM T03691 CUG8R2 44567705 IC50 = 6 nM T03691 C2W1QJ 44567706 IC50 = 46 nM T03691 CW04CP 44567707 IC50 > 1000 nM T03691 CU64DK 44567730 IC50 = 17 nM T03691 C4CT7N 44567731 IC50 = 19 nM T03691 CO34LZ 44567732 IC50 = 5 nM T03691 CCW8D0 44567733 IC50 = 370 nM T03691 CX3G6O 44567767 IC50 = 330 nM T03691 CB56YA 44567768 IC50 = 19 nM T03691 CYC36D 44567769 IC50 = 7 nM T03691 C3IQR6 44567770 IC50 = 15 nM T03691 CZ96EF 44567803 IC50 > 1000 nM T03691 C89ZYK 44567804 IC50 = 44 nM T03691 CE2AQ0 44567832 IC50 = 260 nM T03691 C5W4JA 44567833 IC50 = 160 nM T03691 COY40L 44567834 IC50 = 220 nM T03691 C8SQ4Z 44567868 IC50 = 100 nM T03691 CHU82T 44567909 IC50 = 30 nM T03691 CUS32Z 44567910 IC50 = 3 nM T03691 CW94PM 44567911 IC50 = 130 nM T03691 CM24HC 44567964 IC50 = 3 nM T03691 CL9YI1 44567965 IC50 = 5 nM T03691 CX9LQ3 44567966 IC50 = 11 nM T03691 CEO7P3 44567967 IC50 = 9 nM T03691 CRN2L1 44568006 IC50 = 60 nM T03691 CV2TL8 44568007 IC50 = 2 nM T03691 C2OYI8 44568008 IC50 = 7 nM T03691 CC0MY4 44568009 IC50 = 15 nM T03691 CF1G0U 44568042 IC50 = 5 nM T03691 CHK8A9 44568043 IC50 = 1 nM T03691 CQF40E 44568044 IC50 = 20 nM T03691 C4HAL0 44568086 IC50 = 6 nM T03691 CP5Y7Z 44568087 IC50 = 870 nM T03691 CPM15D 44568088 IC50 = 40 nM T03691 CPQ0B3 44568089 IC50 = 6 nM T03691 C79VML 44568117 IC50 = 350 nM T03691 CR95HI 44568118 IC50 = 1500 nM T03691 CO86KD 44568119 IC50 = 18 nM T03691 CWO79X 44568125 IC50 = 23 nM T03691 CER6N1 44568126 IC50 = 13 nM T03691 CI4O6Q 44568127 IC50 = 4 nM T03691 C0S1DK 44568156 IC50 = 25 nM T03691 C7CV0P 44568157 IC50 = 7 nM T03691 C7WHV5 44568158 IC50 = 290 nM T03691 CJI96U 44568159 IC50 = 6 nM T03691 C5N1LX 44568161 IC50 = 19 nM T03691 C5FH8Q 44568162 IC50 = 5 nM T03691 C1HBE5 44568163 IC50 = 9 nM T03691 CTP61K 44593514 IC50 = 60 nM T03691 CDA52G 44593517 IC50 = 16 nM T03691 CT7E4Q 44593519 IC50 = 60 nM T03691 CBF04L 44593520 IC50 = 57 nM T03691 CIC46F 44818806 IC50 = 4 nM T03691 C1C4UK 46861647 IC50 = 23 nM T03691 C0SJ9C 46888102 IC50 = 29 nM T03691 C2EA5M 46888103 IC50 = 114 nM T03691 C8EGX0 46888144 IC50 = 93 nM T03691 CH7E0F 46888145 IC50 = 174 nM T03691 C9JP5S 46888146 IC50 = 315 nM T03691 COC43S 46888147 IC50 = 438 nM T03691 C4ZK6A 46888148 IC50 = 40 nM T03691 CA4E8K 46888149 IC50 = 880 nM T03691 CPD65I 46888189 IC50 = 212 nM T03691 CD20GA 46888190 IC50 = 53 nM T03691 CJ08AD 46888191 IC50 = 6900 nM T03691 CYP63X 46888192 IC50 = 56 nM T03691 C49EUC 46888239 IC50 = 60 nM T03691 CVCN63 46888240 IC50 = 93 nM T03691 C0HT6A 46888241 IC50 = 6 nM T03691 CA7EF5 46888242 IC50 = 660 nM T03691 C78XZV 49804917 IC50 = 680 nM T03691 CEHY29 49804918 IC50 = 470 nM T03691 C6IWU7 49804919 IC50 = 370 nM T03691 C8W3GR 49804920 IC50 > 100000 nM T03691 CQO37H 49805049 IC50 = 180 nM T03691 CQD83P 49805050 IC50 = 580 nM T03691 CC51BP 49805051 IC50 > 100000 nM T03691 C5L4CW 49805052 IC50 > 100000 nM T03691 C8JVU3 49805053 IC50 > 100000 nM T03691 C8XY3D 49805054 IC50 > 100000 nM T03691 C5MDK8 49805055 IC50 = 4300 nM T03691 C51KQC 49805174 IC50 = 2500 nM T03691 C8CER6 49805175 IC50 = 220 nM T03691 C1LGX6 49805176 IC50 = 540 nM T03691 C0HTK6 49805177 IC50 = 2000 nM T03691 CX6K0C 49805178 IC50 = 40 nM T03691 C0S4FY 49805179 IC50 = 290 nM T03691 CD8J0L 49805180 IC50 = 110 nM T03691 CBK9A7 49805302 IC50 = 970 nM T03691 CVD4T1 49805303 IC50 = 29 nM T03691 CU34WJ 49805304 IC50 > 100000 nM T03691 CVI2E6 49805305 IC50 > 100000 nM T03691 CRV4K9 49805306 IC50 = 3400 nM T03691 CLR02I 49805307 IC50 > 100000 nM T03691 C54QKF 49832992 IC50 = 66 nM T03691 CPH98L 49832994 IC50 = 330 nM T03691 C6S0PJ 49834281 IC50 = 26 nM T03691 CB14NH 49834447 IC50 = 67 nM T03691 CW2X3D 53230825 IC50 = 300 nM T03691 C96ONX 53230826 IC50 = 1800 nM T03691 C48JHC 53320960 IC50 > 1000000 nM T03691 CO0X3H 53324937 IC50 > 1000000 nM T03691 C8FSZ5 54580778 IC50 = 5 nM T03691 CZV9R1 54585654 IC50 = 9 nM T03691 C54JSK 57448273 IC50 = 16 nM T03691 CVNR58 57448274 IC50 = 6 nM T03691 C5CBG4 57448276 IC50 = 14 nM T03691 CUWK92 57448281 IC50 = 11 nM T03691 CY86DR 57448284 IC50 = 6 nM T03691 C74GKR 57448289 IC50 = 29 nM T03691 CPMK57 57448305 IC50 = 1800 nM T03691 CVJ9H0 57448310 IC50 = 614 nM T03691 CAE6B5 57448332 IC50 = 8 nM T03691 CK9TD7 57448346 IC50 = 40 nM T03691 CA6YR3 57448356 IC50 = 3 nM T03691 C0I1CB 57448358 IC50 = 6 nM T03691 CB47MQ 57514846 IC50 = 5 nM T03691 CEQ1P7 59577373 IC50 = 430 nM T03691 C6LO9D 59577386 IC50 = 3.7 nM T03691 C5YNO0 59577401 IC50 = 1.6 nM T03691 C0MRI9 59577413 IC50 = 7 nM T03691 C81YWC 59577483 IC50 = 62 nM T03691 C4M0FX 59577537 IC50 = 340 nM T03691 CGA07I 59577546 IC50 = 14 nM T03691 C49TRA 59577564 IC50 = 4.6 nM T03691 C5U7XF 59577577 IC50 = 2370 nM T03691 C3LT1F 59577582 IC50 = 140 nM T03691 CP6S7R 59577589 IC50 = 340 nM T03691 C6DTM9 59577598 IC50 = 25 nM T03691 CIPH56 59577613 IC50 = 58 nM T03691 CEP3R7 59577628 IC50 = 51 nM T03691 CH1R5P 59577638 IC50 = 7.3 nM T03691 C7EH8Z 59577658 IC50 = 2130 nM T03691 CTK3V4 59577695 IC50 = 340 nM T03691 CB94OG 59577703 IC50 = 7.3 nM T03691 CB15GI 59577729 IC50 = 3 nM T03691 CU5VA6 59577731 IC50 = 300 nM T03691 CT28XN 59577737 IC50 = 8.3 nM T03691 CQIV90 59871873 IC50 = 8900 nM T03691 CFRD26 66559288 Ki > 100000 nM T03691 CRYF85 66560595 Ki > 1000000 nM T03691 CDRP79 66560597 Ki > 100000 nM T03691 C3Q0GW 66560599 Ki = 470000 nM T03691 CC9YW6 66560603 Ki > 100000 nM T03691 CT0NH8 66560605 Ki > 100000 nM T03691 CS12OR 66560607 Ki > 100000 nM T03691 CLZ3A5 66787400 IC50 = 34 nM T03691 CK43VF 66787512 IC50 = 7.3 nM T03691 CV6Z2X 67204288 IC50 = 7 nM T03691 C3WJ5C 67260498 IC50 = 14 nM T03691 C0FPX9 71391212 IC50 > 100000 nM T03691 CU3KE8 71453804 Ki > 1000000 nM T03691 C6VDY5 71456055 IC50 = 0.3 nM T03691 C1NH9X 71457850 IC50 = 1 nM T03691 C3KF2D 71459164 Ki > 100000 nM T03691 CBSY93 71461487 IC50 = 4 nM T03691 CL8T6O 71568931 IC50 = 30000 nM T03691 CP5AU8 71568933 IC50 = 1300 nM T03691 CVE35U 71568934 IC50 = 41800 nM T03691 CGIA28 71569090 IC50 = 6800 nM T03691 C8HL5R 71716159 IC50 = 5200 nM T03691 CH5WJ9 71716778 IC50 = 670 nM T03691 C9IHB6 71717381 IC50 = 5800 nM T03691 CX48SM 71717980 IC50 = 9270 nM T03691 CUD01L 71719202 IC50 = 3800 nM T03691 CT74WK 71720417 IC50 = 9900 nM T03691 C0HSC8 73346520 Ki = 1640 nM T03691 C8SD9P 73346521 Ki = 8650 nM T03691 CGZ6Y8 73346522 Ki = 1060 nM T03691 C43IPQ 73348006 Ki = 172 nM T03691 CS9C0W 73351108 Ki = 369 nM T03691 C27JUH 73352576 Ki = 607 nM T03691 CVP03Z 73352577 Ki = 629 nM T03691 CDAB86 73354065 Ki = 4290 nM T03691 CK3Z8U 73354066 Ki = 643 nM T03691 C92DXZ 73354067 Ki = 3560 nM T03691 CCI18Y 73355591 Ki = 93 nM T03691 CRX8A0 73355592 Ki = 2590 nM T03691 CQB1P2 87057595 IC50 = 60 nM T03691 CR8M9J 91721066 IC50 = 4920 nM T03691 CJA5U6 91721119 IC50 > 100000 nM T03691 C0UJL2 101621289 IC50 = 29470 nM T03691 CC87OM 132547282 IC50 = 3010 nM T03691 CJXP43 134129959 IC50 = 56270 nM T03691 C96ATO 134130173 IC50 = 45610 nM T03691 CFQ65A 134130915 IC50 = 77820 nM T03691 C79YFW 134131352 IC50 > 100000 nM T03691 CSH73J 138756786 IC50 = 200 nM T03691 CP5A1Q 141624077 Ki = 5.3 nM T03691 C86VOP 145704648 IC50 = 13900 nM T03691 C38IXU 145966119 IC50 = 8 nM T03691 CVX5E1 155512701 IC50 = 8350 nM T03691 C7FMD1 155513489 IC50 = 900 nM T03691 C8OGV6 155514713 IC50 > 30000 nM T03691 CJPY40 155521682 IC50 > 30000 nM T03691 C01EFS 155528719 IC50 = 400 nM T03691 CF6AC7 155530648 IC50 > 30000 nM T03691 CQF20U 155535260 IC50 = 240 nM T03691 CA2V8K 155537914 IC50 = 260 nM T03691 C6D0IZ 155545668 IC50 = 200 nM T03691 C9UO2J 155546182 IC50 = 210 nM T03691 CLAU71 155546998 IC50 = 100 nM T03691 CJES98 155548156 IC50 = 230 nM T03691 CRW78E 155548442 IC50 > 30000 nM T03691 CHE69M 155553765 IC50 = 3800 nM T03691 C24EVD 155554682 IC50 > 30000 nM T03691 CBK06N 155557826 Ki = 4.6 nM T03691 CED94J 155563098 IC50 > 30000 nM T03691 CVY1U7 155564021 IC50 > 30000 nM T03691 C10XMH 155564211 IC50 = 1200 nM T03691 D00EJS 16054 IC50 > 1000000 nM T03691 D00FCJ 24901626 IC50 = 150 nM T03691 D00FDS 29293603 IC50 = 126 nM T03691 D00TNN 45253769 IC50 = 207 nM T03691 D00TWK 185914 IC50 = 145000 nM T03691 D00UIN 11739248 IC50 = 11 nM T03691 D01KOI 346926 IC50 > 1000000 nM T03691 D01QWO 44562814 IC50 = 5560 nM T03691 D01RVF 44129620 IC50 = 157 nM T03691 D01YJJ 24901620 IC50 = 31 nM T03691 D02AYI 11031651 IC50 = 228 nM T03691 D02TMR 24901614 IC50 = 2600 nM T03691 D03GON 11416868 IC50 = 4 nM T03691 D04CZF 24901607 IC50 = 23 nM T03691 D04DRM 24901601 IC50 = 7200 nM T03691 D04KQF 6675804 IC50 > 10000 nM T03691 D04QJY 123982 IC50 = 5 nM T03691 D04ZLZ 24901603 IC50 = 1100 nM T03691 D05NXQ 29293599 IC50 = 44 nM T03691 D06RWH 22690393 IC50 = 135 nM T03691 D06SMN 16222640 IC50 = 87 nM T03691 D07KBF 24901625 IC50 = 2800 nM T03691 D07LTR 21883856 IC50 = 4130 nM T03691 D07TVA 44562812 IC50 = 5720 nM T03691 D07ZJS 46888070 IC50 = 105 nM T03691 D08TNQ 24768560 IC50 = 20 nM T03691 D08UIO 11257168 IC50 = 66 nM T03691 D08WZB 24901612 IC50 = 9700 nM T03691 D09BWE 11473281 IC50 = 34 nM T03691 D09DRF 90334 IC50 = 308000 nM T03691 D09MDO 22692237 IC50 = 61 nM T03691 D09OWF 24901615 IC50 = 19 nM T03691 D09PGC 24901582 IC50 = 58 nM T03691 D0A2YG 7060565 IC50 = 1077000 nM T03691 D0B0DP 24901630 IC50 = 6 nM T03691 D0B9UW 24901629 IC50 = 29 nM T03691 D0C1XE 46888101 IC50 = 60 nM T03691 D0C8MT 260806 IC50 = 12500 nM T03691 D0DI4I 24901621 IC50 = 18 nM T03691 D0G0JC 1082702 IC50 = 1321000 nM T03691 D0G8SW 24901627 IC50 = 13 nM T03691 D0H9NZ 46888243 IC50 = 342 nM T03691 D0HA1K 24901600 IC50 = 680 nM T03691 D0I4OV 2776332 IC50 = 98000 nM T03691 D0I7MC 44562857 IC50 = 2480 nM T03691 D0J0WO 7023019 IC50 = 3673000 nM T03691 D0LZ3O 24768559 IC50 = 5400 nM T03691 D0M2CY 24901637 IC50 = 21 nM T03691 D0N6TC 24901619 IC50 = 46 nM T03691 D0P7DF 16039611 IC50 = 340 nM T03691 D0PF9Q 11472798 IC50 = 59 nM T03691 D0Q8LS 11427736 IC50 = 17 nM T03691 D0R5HK 16760703 IC50 > 10000 nM T03691 D0R7BT 2776424 IC50 = 38900 nM T03691 D0SZ9E 177363 IC50 = 570 nM T03691 D0U1EV 24901604 IC50 = 1600 nM T03691 D0U1UV 24901602 IC50 = 9300 nM T03691 D0U2AM 24901616 IC50 = 21 nM T03691 D0V0MH 3017356 IC50 = 1.4 nM T03691 D0VN8V 44818625 IC50 = 8700 nM T03691 D0W2OP 10609349 IC50 = 280 nM T03691 D0Y6IV 44562813 IC50 = 5690 nM T03691 D0Z6DL 24901617 IC50 = 210 nM T66935 CD1Q4C 2331 IC50 > 1000000 nM T66935 CWB45K 482198 IC50 = 22000 nM T66935 CAKC37 873742 EC50 > 150000 nM T66935 C3V8NS 1258015 EC50 = 11000 nM T66935 CRM4I5 1517285 EC50 > 150000 nM T66935 CQP51Z 2829333 EC50 = 30000 nM T66935 CK24BY 3014425 IC50 = 500000 nM T66935 CQ95WV 3870576 EC50 > 50000 nM T66935 C8KZ7C 4093912 EC50 = 140000 nM T66935 CG36WM 5300082 EC50 = 57000 nM T66935 C0IS9F 6324454 EC50 = 50000 nM T66935 CW9FY1 6918639 IC50 = 120 nM T66935 CTRZ81 7113016 EC50 > 30000 nM T66935 C6UIL3 7122772 EC50 > 150000 nM T66935 CO16NI 7164286 EC50 > 150000 nM T66935 CV4YK1 16832109 EC50 = 110000 nM T66935 CO92DI 46361427 EC50 = 110000 nM T66935 CKX0Z7 53387188 IC50 = 12000 nM T66935 CD5HO1 53391538 IC50 = 42000 nM T66935 CWP5D9 53391539 IC50 = 27000 nM T66935 C3EQY1 53391540 IC50 = 21000 nM T66935 CY4KI9 53391541 IC50 = 25000 nM T66935 C4V3LQ 53391542 IC50 = 26000 nM T66935 C0YT2O 53391636 IC50 = 61000 nM T66935 C52QIC 53392780 IC50 = 140000 nM T66935 CQV9P5 53392959 IC50 = 500000 nM T66935 C3RS9C 53392960 IC50 = 117000 nM T66935 C40EKO 53392961 IC50 = 61000 nM T66935 C1S3NU 56658116 IC50 = 26000 nM T66935 C3IGF0 56658117 IC50 = 72000 nM T66935 CV8B2N 56665040 IC50 = 8000 nM T66935 C1RC6I 76850155 EC50 > 70000 nM T66935 CP30IO 121398087 EC50 = 5200 nM T66935 CC64BH 121398103 EC50 = 480 nM T66935 CR9WM2 121398113 EC50 = 620 nM T66935 C7J5XW 121398163 EC50 = 2300 nM T66935 C3XY8F 121398171 EC50 = 2100 nM T66935 C12GMC 121398173 EC50 = 1800 nM T66935 C59LIE 121398178 EC50 = 29 nM T66935 CDCJ30 121398201 EC50 = 5000 nM T66935 CO49WL 121398202 EC50 = 64 nM T66935 CA09EU 121398203 EC50 = 860 nM T66935 CV2B8D 121398243 EC50 = 1600 nM T66935 C79MTN 121398248 EC50 = 19 nM T66935 CS52JD 121398291 EC50 = 120 nM T66935 CML3I9 121398292 EC50 = 45 nM T66935 C6RB7G 121398298 EC50 = 1200 nM T66935 CEML83 121398299 EC50 = 1700 nM T66935 CH8B0N 121398301 EC50 = 1100 nM T66935 C4EW9G 121398347 IC50 = 290 nM T66935 CHB8V4 121398349 EC50 = 2800 nM T66935 CO7PY4 121398362 EC50 = 280 nM T66935 CKY2M9 121398376 EC50 = 380 nM T66935 CLE59U 121398379 EC50 = 3000 nM T66935 C1CAZ2 121398391 EC50 = 470 nM T66935 C4CPO3 121398401 EC50 = 280 nM T66935 CQ2P0I 121398419 EC50 = 3000 nM T66935 C1LBA9 121398427 EC50 = 450 nM T66935 C4YCA0 121398429 EC50 = 270 nM T66935 CK28VL 121398451 EC50 = 2500 nM T66935 C0RNY4 121398470 EC50 = 250 nM T66935 C1C4ZJ 121398471 EC50 = 1100 nM T66935 CB7EY8 121398481 EC50 = 2700 nM T66935 C6NC0J 121398483 EC50 = 250 nM T66935 CRGV62 121398484 EC50 = 3200 nM T66935 CLZ1D4 121398509 EC50 = 440 nM T66935 CQE7J0 121398517 IC50 = 80 nM T66935 C5JYP2 121398518 EC50 = 49 nM T66935 CRQ92F 121398519 EC50 = 450 nM T66935 CR3PS6 121398524 EC50 = 1300 nM T66935 CU8H1R 121398529 EC50 = 910 nM T66935 CWV73S 121398540 EC50 = 390 nM T66935 CY9T6E 121398541 EC50 = 380 nM T66935 C9JT4U 121398546 EC50 = 560 nM T66935 CX8NR3 121398556 EC50 = 52 nM T66935 CGT19I 121398625 EC50 = 2400 nM T66935 CRIH72 121398630 EC50 = 23 nM T66935 CHE72W 121398637 EC50 = 76 nM T66935 C43HAR 121398640 EC50 = 1200 nM T66935 C8H7MG 121398649 EC50 = 4000 nM T66935 CQW92J 121398660 EC50 = 5200 nM T66935 C59ORZ 121398668 EC50 = 69 nM T66935 CGKV70 121398676 EC50 = 370 nM T66935 CTX87P 121398678 EC50 = 4000 nM T66935 CNS8F3 121398699 EC50 = 3100 nM T66935 CVO51J 121398702 EC50 = 5000 nM T66935 CV8FO5 121398710 EC50 = 4600 nM T66935 CK06SA 121398719 EC50 = 5800 nM T66935 C8HV4N 121398731 EC50 = 120 nM T66935 CTWU21 121398732 EC50 = 78 nM T66935 CG72EA 121398751 EC50 = 180 nM T66935 CZ7BW5 121398752 EC50 = 4000 nM T66935 C6U8PC 121398766 EC50 = 26 nM T66935 C2Z4ML 121398777 EC50 = 1800 nM T66935 CBE60D 121398796 EC50 = 1200 nM T66935 C6UJ5E 121398814 EC50 = 3200 nM T66935 CE6GB0 121398817 EC50 = 1300 nM T66935 C41TRQ 121398822 EC50 = 1300 nM T66935 CX4P0U 121398824 EC50 = 7000 nM T66935 C32APX 121398861 EC50 = 8000 nM T66935 CP0RB2 121398889 EC50 = 2000 nM T66935 CY76IA 121398901 EC50 = 38 nM T66935 COXV78 121404613 EC50 = 6000 nM T66935 C23VRS 121404646 EC50 = 770 nM T66935 C84VZN 134169659 EC50 = 1800 nM T66935 CR08FV 134169675 EC50 = 1100 nM T66935 C36UOG 134169680 EC50 = 1400 nM T66935 C2OKH4 134169681 EC50 = 530 nM T66935 CD8R9P 134169682 EC50 = 1600 nM T66935 C7NZ3O 134169687 EC50 = 480 nM T66935 CU0P1A 134169689 EC50 = 4100 nM T66935 CB7XR1 134169693 EC50 = 3300 nM T66935 CH89LT 134169694 EC50 = 4.8 nM T66935 C7AVY0 134169696 EC50 = 6 nM T66935 CQ78WB 134169699 EC50 = 470 nM T66935 C6YOM2 134169705 EC50 = 880 nM T66935 CO2LF4 145980040 EC50 = 16000 nM T66935 C7J3IZ 145980728 EC50 = 24000 nM T66935 C61LYK 145981066 EC50 = 20000 nM T66935 CU2D0Z 145981393 EC50 > 150000 nM T66935 CNM1G6 145981912 EC50 = 110000 nM T66935 C70IMH 145982111 EC50 > 150000 nM T66935 C95GPH 145983675 EC50 = 3300 nM T66935 C35NLD 145985394 EC50 = 13000 nM T66935 CER3G0 145987067 EC50 = 10000 nM T66935 CRUO60 145988794 EC50 = 12000 nM T66935 C6X5VM 145990022 EC50 = 26000 nM T66935 CG08AY 145990890 EC50 = 13000 nM T66935 C7ZW1B 145991145 EC50 > 150000 nM T66935 C8MXN4 145991355 EC50 = 88000 nM T66935 C2EA0L 145991422 EC50 = 23000 nM T66935 CXQ20E 145992505 EC50 = 12000 nM T66935 C43PCI 145993165 EC50 > 150000 nM T66935 C75SXJ 145993230 EC50 = 6000 nM T66935 CT1Y6Z 145993252 EC50 = 21000 nM T66935 C8U9NF 145993965 EC50 = 49000 nM T66935 CR7Z8P 145994151 EC50 > 150000 nM T66935 C5IR1N 155521896 IC50 = 3600 nM T66935 C0GW8L 155526220 IC50 = 320 nM T66935 C5B2WP 155526343 IC50 = 30 nM T66935 C8PD4L 155527387 IC50 = 20 nM T66935 CFY91Q 155541426 IC50 = 90 nM T66935 CIU95N 155556583 IC50 = 1520 nM T81452 D0T9TJ 3034010 IC50 = 13.18 nM T81452 D0CW8S 71657619 IC50 = 253 nM T81452 CQP8H6 53364459 IC50 = 39.81 nM T81452 C5U3CY 53364540 IC50 = 39.81 nM T81452 CS64LM 57519635 IC50 = 19.95 nM T81452 CYO64A 71656315 IC50 = 2100 nM T81452 C50OAM 71656796 IC50 = 600 nM T81452 C2TO5C 71656797 IC50 > 10000 nM T81452 CN89IX 71656798 IC50 = 91 nM T81452 C49OFR 71656799 IC50 = 182 nM T81452 C92YGU 71657082 IC50 = 190 nM T81452 CV5PM2 71657185 IC50 = 1800 nM T81452 CPT0H5 71657290 IC50 = 3000 nM T81452 CM2ZB8 71657292 IC50 = 1300 nM T81452 CBSW63 71657395 IC50 = 1300 nM T81452 CVUD47 71657398 IC50 > 10000 nM T81452 C2KHF7 89677087 IC50 = 3400 nM T81452 CXT5C7 89682527 IC50 = 3800 nM T81452 CPF01Q 89682653 IC50 = 290 nM T81452 CN8HX3 89682683 IC50 = 2500 nM T81452 CY7PD2 89682704 IC50 = 170 nM T81452 CNU8L7 89682719 IC50 = 130 nM T81452 CUJ4Q7 97289144 IC50 = 630.96 nM T81452 CA0B1S 97289145 IC50 = 2.512 nM T81452 C5DP6A 102340761 Ki = 800 nM T81452 CFVX28 102596130 IC50 = 1778.28 nM T81452 C1LD8T 118709692 Ki = 18300 nM T81452 C7WM1Y 118709694 Ki = 2700 nM T81452 CFTM51 118729369 IC50 = 750 nM T81452 CY9UH3 121513897 IC50 = 43.65 nM T81452 CJ1GQ9 122188643 IC50 = 216 nM T81452 CYZN76 122188783 IC50 = 130 nM T81452 C0Y9DJ 122188784 IC50 = 73 nM T81452 COT9L7 122189215 IC50 = 446.68 nM T81452 CUB13M 122189217 IC50 = 870 nM T81452 C7JU5Q 122530045 IC50 = 2100 nM T81452 CEA48I 129188688 IC50 = 2.512 nM T81452 CU0D3S 130346049 IC50 = 660 nM T81452 CW1G0V 134131835 IC50 = 3162.28 nM T81452 C2PYB4 134133861 IC50 = 158.49 nM T81452 CM4WT3 134133947 IC50 = 39.81 nM T81452 CS6VC7 134134749 IC50 = 251.19 nM T81452 C8NST5 134135610 IC50 = 251.19 nM T81452 CZW3T0 134138122 IC50 = 7943.28 nM T81452 C2GX1J 134138767 IC50 = 39.81 nM T81452 CK7MS5 134139434 IC50 = 199.53 nM T81452 CTWL68 134140363 IC50 = 125.89 nM T81452 C3BWS0 134141954 IC50 > 10000 nM T81452 CWES31 134142232 IC50 = 50.12 nM T81452 CBA6M0 134142396 IC50 = 199.53 nM T81452 C4H7UW 134143500 IC50 = 158.49 nM T81452 CYI16B 134145542 IC50 = 158.49 nM T81452 CCBN29 134147523 IC50 = 3162.28 nM T81452 CMQ9L3 134150114 IC50 = 2511.89 nM T81452 CU7D8C 134151520 IC50 > 10000 nM T81452 C2N3VI 134153875 IC50 = 25.12 nM T81452 CXYP40 134156008 IC50 = 3162.28 nM T81452 CSOX06 134156265 IC50 = 251.19 nM T81452 CKJ1X4 134157652 IC50 = 199.53 nM T81452 CZ3F5D 135239539 IC50 = 562 nM T81452 C0U9TO 137546866 IC50 = 5300 nM T81452 CWZ92Q 137651267 IC50 = 7100 nM T81452 CB8IM1 138319671 IC50 > 10000 nM T81452 C5XM3H 145949852 IC50 > 10000 nM T81452 CSM7J0 145951205 IC50 > 10000 nM T81452 C4IX1W 145951504 IC50 > 10000 nM T81452 C06VUY 145951905 IC50 = 530 nM T81452 CV0S3L 145953742 IC50 = 3000 nM T81452 C2KJ8F 145955689 IC50 > 10000 nM T81452 C46LCZ 145955918 IC50 > 10000 nM T81452 CP0L8K 145956576 IC50 > 10000 nM T81452 CEX3U4 145956825 IC50 > 10000 nM T81452 CX70KY 145957108 IC50 > 10000 nM T81452 CDEK59 145959588 IC50 > 10000 nM T81452 CDN40B 145972411 IC50 > 10000 nM T81452 CO1MF8 145979117 IC50 = 10 nM T81452 CBF8Z1 145979505 IC50 = 12.59 nM T81452 CPJ13H 145980248 IC50 = 251.19 nM T81452 CZ5GX0 145980541 IC50 = 2.512 nM T81452 C9ZVP4 145980767 IC50 = 3.162 nM T81452 C4CW1J 145981620 IC50 = 794.33 nM T81452 CD5G1L 145982097 IC50 > 10000 nM T81452 C0T9PD 145982431 IC50 = 31.62 nM T81452 C9XUQ0 145983194 IC50 > 10000 nM T81452 C3IA4D 145986832 IC50 = 5.012 nM T81452 C8U1LO 145987585 IC50 = 25.12 nM T81452 CAH95K 145988033 IC50 = 316.23 nM T81452 CV1IH0 145988362 IC50 > 10000 nM T81452 CSTI30 145988650 IC50 = 100 nM T81452 CU1BT5 145989121 IC50 > 10000 nM T81452 CT0H4P 145990805 IC50 = 6.31 nM T81452 C1Z9EW 145990933 IC50 = 3.162 nM T81452 C0ULZ5 145990999 IC50 > 10000 nM T81452 C3OXW0 145992126 IC50 > 10000 nM T81452 C3JMC7 145992455 IC50 > 10000 nM T81452 C4Q1ME 145992746 IC50 = 158.49 nM T81452 CXYG34 145993594 IC50 > 10000 nM T81452 CO67DP 145994122 IC50 = 15.85 nM T81452 CEQ7G4 155510849 IC50 = 2500 nM T81452 C9CD3Q 155511585 IC50 = 99 nM T81452 C25OAR 155512542 IC50 = 540 nM T81452 CI2WL8 155513853 IC50 = 1500 nM T81452 CBG4Q8 155521008 IC50 = 5300 nM T81452 CL6Z1R 155526799 IC50 = 1100 nM T81452 C6Z9GK 155531741 IC50 > 10000 nM T81452 CW7N6K 155533489 IC50 = 2700 nM T81452 CQ67EK 155543660 IC50 = 940 nM T81452 C8XZ7V 155545255 IC50 = 1400 nM T81452 C9WGK1 155547201 IC50 = 10000 nM T81452 C6TPM9 155549206 IC50 > 10000 nM T81452 CH78YM 155549832 IC50 = 1600 nM T81452 C4U9WO 155550747 IC50 = 5000 nM T81452 CY52RZ 155560863 IC50 > 10000 nM T73342 D0HP3M 513004 EC50 = 3100 nM T73342 C0N8AB 512986 IC50 = 58000 nM T73342 C0PB1Y 512989 IC50 = 860 nM T73342 CN1R9O 512990 IC50 = 880 nM T73342 CD20ZM 512991 IC50 = 24 nM T73342 C8XJW6 512992 IC50 = 4000 nM T73342 CN2F5R 512993 IC50 = 180 nM T73342 CM9EX7 512994 IC50 = 860 nM T73342 CNL2B0 512995 IC50 = 11000 nM T73342 CJH3E1 512996 IC50 = 22 nM T73342 CBK0S8 512997 IC50 = 340 nM T73342 CK1J4A 512999 IC50 = 115000 nM T73342 CWD95K 513001 IC50 = 36 nM T73342 C05URV 513002 IC50 = 22 nM T73342 CI3D9Z 513003 EC50 = 30000 nM T73342 CQK80X 513005 EC50 = 35000 nM T73342 CVD10B 513006 EC50 = 7300 nM T73342 C1TZD5 513007 EC50 = 30000 nM T73342 C03DUB 513008 EC50 = 150000 nM T73342 C2N8BE 513009 EC50 = 6500 nM T73342 C8UJ7P 513010 EC50 = 12000 nM T73342 COB6C7 513011 IC50 = 0.7 nM T73342 CI8QD0 513012 IC50 = 7.5 nM T73342 CRYB30 513013 IC50 = 4 nM T73342 C5AHP9 513014 IC50 = 1 nM T73342 CE8UQ1 513015 IC50 = 5 nM T73342 C90KIJ 513016 IC50 = 34 nM T73342 C3GU9T 515251 IC50 = 15 nM T73342 CIJC18 515252 IC50 = 440 nM T73342 CK58FD 515254 IC50 = 7 nM T73342 CO45XM 515255 IC50 = 3 nM T73342 CBO59N 515256 IC50 = 2200 nM T73342 CXP13E 515257 IC50 = 7000 nM T73342 C9EU0J 515258 IC50 = 3500 nM T73342 C6XRA1 515272 IC50 = 500 nM T73342 CE3FP7 515277 IC50 = 0.6 nM T73342 CC5KE7 515278 IC50 = 6 nM T73342 CGYO68 515279 IC50 = 100 nM T73342 C8P2LI 515280 IC50 = 350 nM T73342 C5BVI1 515281 IC50 = 40 nM T73342 C8ENO3 515282 IC50 = 1900 nM T73342 CCIH63 515283 IC50 = 27 nM T73342 C2IBC5 515284 IC50 = 18 nM T73342 C5H4PL 515285 IC50 = 2700 nM T73342 CB3CA2 515286 IC50 = 2000 nM T73342 C8LC5F 515287 IC50 = 7 nM T73342 C8HW5T 515288 IC50 = 3 nM T73342 CMC61D 515289 IC50 = 5 nM T73342 CH2C5Y 515343 IC50 = 760000 nM T73342 CTW72N 515370 IC50 = 43 nM T73342 C8RF7H 5274922 IC50 = 25000 nM T73342 CTR8V7 5274931 IC50 = 15000 nM T73342 CC4UB1 5496256 IC50 = 8800 nM T73342 CU4WD1 5496499 IC50 = 13300 nM T73342 C5T9FB 7075199 IC50 = 232000 nM T73342 C9OFU4 10079737 IC50 = 1900 nM T73342 CAUH90 10463141 IC50 = 20000 nM T73342 CI75GJ 11693485 IC50 = 40000 nM T73342 C4FT7Z 14861763 Ki = 830000 nM T73342 CYT06R 44272984 IC50 = 5000 nM T73342 CUA50V 44272989 IC50 = 12000 nM T73342 CEAM73 44273125 IC50 = 6000 nM T73342 C7Y6RA 44273175 IC50 = 600000 nM T73342 C4BMN3 44346525 IC50 = 6.4 nM T73342 C4HYV6 44350302 IC50 = 412000 nM T73342 CG86EB 44350389 IC50 > 400000 nM T73342 CDZ4Y6 44395455 IC50 = 2400 nM T73342 C1P0SZ 44395456 IC50 = 2400 nM T73342 CU97LO 44395457 IC50 = 22000 nM T73342 CGW91B 49799941 IC50 = 55 nM T73342 C9G2RP 56657765 IC50 > 400000 nM T73342 C0T1LH 56657837 IC50 = 61 nM T73342 C7Q9EV 56657845 IC50 > 400000 nM T73342 CQ3E7K 56664763 IC50 = 100000 nM T73342 CRI89Z 56664822 IC50 > 400000 nM T73342 C5I0HN 56664823 IC50 = 100000 nM T73342 CRF08D 56668183 IC50 = 500000 nM T73342 CFA5X6 56675073 IC50 = 30000 nM T73342 C3ON8X 56675131 IC50 = 28000 nM T73342 CG94JM 56675133 IC50 > 400000 nM T73342 CB4O3H 56675162 IC50 = 11000 nM T73342 CT46FB 56678438 IC50 = 80000 nM T73342 C2V6MO 56681722 IC50 = 322000 nM T73342 C0H6SU 56681723 IC50 = 207000 nM T73342 CDG54O 135521627 IC50 = 41591.06 nM T73342 C6UDW4 135559909 IC50 = 14190.58 nM T73342 CJ6NM4 135560361 IC50 = 242102.9 nM T73342 C2S4HO 135612469 IC50 = 39264.49 nM T73342 C80LSM 135659447 IC50 = 287078.06 nM T73342 CV74OX 135827898 IC50 = 36475.39 nM T73342 CRB86C 136045853 IC50 = 46773.51 nM T73342 CP1Q4H 136045854 IC50 = 29308.93 nM T73342 CA87HZ 136045855 IC50 = 30408.85 nM T73342 CIA98S 136045856 IC50 = 45081.67 nM T73342 C5VDZ2 136045857 IC50 = 29308.93 nM T73342 C8C0KW 136045858 IC50 = 28575.91 nM T73342 C2JDI7 136045859 IC50 = 43251.38 nM T87023 D06ABF 3957 IC50 = 135000 nM T87023 D0B7NG 2725 IC50 > 50000 nM T87023 D0N7AD 19861 IC50 > 50000 nM T87023 D0S1CQ 133017 IC50 = 3700 nM T87023 D0C2HI 60680 IC50 = 610 nM T87023 D0D5ZV 6918268 IC50 = 10 nM T87023 D0I0UE 9804204 Ki = 0.38 nM T87023 D0P1YE 9852175 Ki = 2270 nM T87023 D01RFI 6439060 IC50 = 40 nM T87023 D05KQE 131925 Ki = 3.2 nM T87023 D07SGB 9830503 Ki = 0.98 nM T87023 D0BD3U 159547 IC50 = 60 nM T87023 D0CB8W 65889 IC50 = 40 nM T87023 D0S4JY 60775 IC50 = 13 nM T87023 CK7G2V 2451 IC50 = 300 nM T87023 C1LF4I 145955 IC50 = 3500 nM T87023 C5EZD4 154087 Ki = 0.57 nM T87023 CN8W3L 197443 Ki = 1.85 nM T87023 C0S9KD 524022 IC50 = 1400 nM T87023 CTJ8V3 5312127 Ki = 9 nM T87023 C4SWU6 6324617 IC50 = 128 nM T87023 C65HYP 9801987 IC50 = 7500 nM T87023 CV14NA 9820228 IC50 = 120 nM T87023 CF24BG 9824829 IC50 = 10 nM T87023 C8PM1J 9862913 IC50 = 150 nM T87023 CQ4LC2 9872676 Ki = 1060 nM T87023 CZ10BK 9936894 IC50 = 33 nM T87023 CZP08M 9971461 IC50 = 19000 nM T87023 CP03CZ 9973198 IC50 = 6500 nM T87023 CUPG51 9993602 IC50 = 55000 nM T87023 CND43U 9995815 IC50 = 82000 nM T87023 C4YI8D 9998465 IC50 = 1100 nM T87023 CZJV17 10002808 IC50 = 1 nM T87023 CJIL81 10015480 IC50 = 5400 nM T87023 C0AXH6 10015659 IC50 = 5700 nM T87023 C1M6LN 10021121 IC50 = 9200 nM T87023 C1ZD8T 10021505 IC50 = 1100 nM T87023 CPWO61 10032022 Ki = 2.5 nM T87023 CZQ0S3 10042229 IC50 = 59400 nM T87023 CE01PB 10048859 IC50 = 13100 nM T87023 CYG62S 10060480 IC50 = 11200 nM T87023 CZ1P5B 10060534 IC50 = 47900 nM T87023 C7SIT3 10060780 IC50 = 15200 nM T87023 CU62MP 10063751 IC50 = 22000 nM T87023 C60ZPH 10065779 IC50 = 900 nM T87023 CAS6X3 10066158 IC50 = 2800 nM T87023 CVIR70 10243193 IC50 = 100000 nM T87023 CLG98E 10244542 IC50 = 14200 nM T87023 CNG1I7 10246399 IC50 > 100000 nM T87023 COUE17 10265702 IC50 = 37200 nM T87023 C5F3NH 10314059 IC50 = 3400 nM T87023 C01NIR 10378954 IC50 = 8100 nM T87023 CHT41W 10378955 IC50 = 5400 nM T87023 C1QJD5 10381070 IC50 = 31800 nM T87023 CAJ38M 10394043 Ki = 3 nM T87023 CH7TP9 10423490 IC50 = 6300 nM T87023 C6FU0R 10427163 IC50 = 40400 nM T87023 COD09C 10444655 IC50 = 100000 nM T87023 C6Y8GR 10448393 IC50 = 17000 nM T87023 CVCX82 10470867 IC50 = 19200 nM T87023 C1D7IZ 10508960 IC50 = 22 nM T87023 C2D4ZJ 10532787 IC50 = 21 nM T87023 CQ4F2U 10604738 IC50 = 2 nM T87023 C1IE7X 10624368 IC50 = 10 nM T87023 C8IAZ9 10628536 IC50 = 23 nM T87023 C9W6MS 10628732 IC50 = 285 nM T87023 COU7F6 10652101 IC50 = 167 nM T87023 C0DQ6Y 10668473 IC50 = 2.3 nM T87023 C3TNZ9 10695884 IC50 = 30 nM T87023 C6ZVJ5 10700170 IC50 = 38 nM T87023 CQPC29 10723353 IC50 = 45 nM T87023 C7PT2Q 10723685 IC50 = 25 nM T87023 C0T9YN 10746928 IC50 = 20 nM T87023 CR60GS 10842032 IC50 = 39 nM T87023 CJ90XQ 11450461 IC50 = 1258.93 nM T87023 CSK06X 11724601 IC50 = 2200 nM T87023 C4MS1K 11771535 IC50 = 575.44 nM T87023 CB4WG1 11779704 IC50 = 4000 nM T87023 CCB59A 13457165 IC50 = 21 nM T87023 CO6U0W 13557454 IC50 = 400 nM T87023 CYIN80 13557456 IC50 = 2500 nM T87023 CG1U7I 13557458 IC50 > 1000 nM T87023 CH93FQ 13557460 IC50 = 350 nM T87023 C05FST 13557462 IC50 > 1000 nM T87023 CW98BF 13557466 IC50 = 1300 nM T87023 CGKW06 13557472 IC50 = 500 nM T87023 C2AG1U 13557473 IC50 = 1000 nM T87023 C1X0ZV 13557474 IC50 = 600 nM T87023 C8FUQ7 13557475 IC50 = 1800 nM T87023 C6PO3S 13557476 IC50 = 700 nM T87023 CBF1U7 13557477 IC50 = 1200 nM T87023 C4VSK3 13557479 IC50 = 5000 nM T87023 C6XHY0 13557482 IC50 > 1000 nM T87023 C70OND 13557486 IC50 = 450 nM T87023 CJ1PE4 13557487 IC50 = 200 nM T87023 C6UCY3 13557494 IC50 = 370 nM T87023 CD6LE3 13557495 IC50 = 1000 nM T87023 C7SR9J 13557496 IC50 = 250 nM T87023 CFJ0L8 13557499 IC50 = 100 nM T87023 CT1J5H 13557504 IC50 = 250 nM T87023 CFLI05 13557506 IC50 = 600 nM T87023 CIL47Q 13557507 IC50 = 400 nM T87023 CUP2I7 13557513 IC50 > 1000 nM T87023 C2V8AG 13557522 IC50 > 1000 nM T87023 C8E4PJ 13739736 IC50 = 1200 nM T87023 CT3U1S 13790031 IC50 > 1000 nM T87023 CS0PY3 13790046 IC50 > 1000 nM T87023 C6AT8X 13999746 IC50 > 1000 nM T87023 CX0V9W 13999749 IC50 > 1000 nM T87023 CB93OT 13999751 IC50 > 1000 nM T87023 CV9U5E 14347330 IC50 = 20 nM T87023 C3FP7J 14347332 IC50 = 40 nM T87023 C6ESQ2 14347334 IC50 = 2 nM T87023 C67VQS 14347337 IC50 = 25 nM T87023 C9VS4E 14347338 IC50 = 85 nM T87023 CZ7I4K 14347339 IC50 = 55 nM T87023 C6OAV8 14347340 IC50 = 25 nM T87023 C6PAT4 14347341 IC50 = 60 nM T87023 CG8IQ9 14347344 IC50 = 115 nM T87023 CX0B4P 14347348 IC50 = 170 nM T87023 C8ZDK4 14347349 IC50 = 250 nM T87023 CWZ7C3 14347351 IC50 = 250 nM T87023 CX0S7Y 14347352 IC50 = 275 nM T87023 CP2O4U 14347354 IC50 = 35 nM T87023 C8WX9A 14347355 IC50 = 300 nM T87023 C6OY8M 14347357 IC50 = 65 nM T87023 CS60FT 14347358 IC50 = 200 nM T87023 CC2UE3 14347360 IC50 = 50 nM T87023 CTR5F1 14347362 IC50 = 250 nM T87023 CNE37W 14347364 IC50 = 400 nM T87023 CH8Q2C 14347367 IC50 = 25 nM T87023 CP54IM 14347368 IC50 = 40 nM T87023 C67VLS 14347369 IC50 = 40 nM T87023 C4BW8G 14347370 IC50 = 60 nM T87023 CT78KD 14347373 IC50 = 300 nM T87023 CDH84A 14347379 IC50 = 4 nM T87023 CC36YX 14347380 IC50 = 2 nM T87023 CO2LJ7 14347392 IC50 = 20 nM T87023 C0CO2F 14347393 IC50 = 20 nM T87023 C3A2QC 14347397 IC50 = 40 nM T87023 C23VKX 14347399 IC50 = 40 nM T87023 CY0E4N 14347400 IC50 = 10 nM T87023 C0NU6E 14347403 IC50 = 30 nM T87023 CM2HR9 14347405 IC50 = 25 nM T87023 CVF20L 14347407 IC50 = 30 nM T87023 CD1QC8 14347409 IC50 = 14 nM T87023 CWO6G1 14347411 IC50 = 9 nM T87023 CPI0K3 14347413 IC50 = 5 nM T87023 CR69MO 14347434 IC50 = 10 nM T87023 C97TAI 14347435 IC50 = 250 nM T87023 CIMJ98 14547222 IC50 = 450 nM T87023 CQ8F7V 14547223 IC50 = 100 nM T87023 CJ13QI 14547295 IC50 = 120 nM T87023 C81BUN 14547296 IC50 = 400 nM T87023 CDF4O5 14547297 IC50 = 30 nM T87023 C89IBG 14547299 IC50 = 700 nM T87023 C8BAM5 14547300 IC50 = 250 nM T87023 CV1TH7 14547302 IC50 = 50 nM T87023 C3STN1 14547304 IC50 = 100 nM T87023 CU15PW 14554123 IC50 > 50000 nM T87023 CZQM08 14554127 IC50 = 33000 nM T87023 CJU02M 14554129 IC50 = 2400 nM T87023 C6RA8W 14554138 IC50 = 13000 nM T87023 CO7B3M 14554145 IC50 = 1800 nM T87023 CPYU15 14554146 IC50 = 1000 nM T87023 CCW31Q 14570074 IC50 = 630 nM T87023 C4HMY8 14570078 IC50 = 500 nM T87023 CP3IQ1 14570080 IC50 = 280 nM T87023 CJD70T 14570083 IC50 = 20 nM T87023 CF4G1X 14570085 IC50 = 300 nM T87023 CZ08OQ 14570086 IC50 = 200 nM T87023 C0TCA7 14570087 IC50 = 400 nM T87023 CUP1G9 14570089 IC50 = 15 nM T87023 CHP0A9 14570090 IC50 = 5 nM T87023 CQ6M7R 14570092 IC50 = 50 nM T87023 CO06RM 14570093 IC50 = 200 nM T87023 CHY5N1 14570094 IC50 = 125 nM T87023 CB0U3J 14570095 IC50 = 200 nM T87023 C46ROI 14570097 IC50 = 200 nM T87023 C4K6PL 14570098 IC50 = 220 nM T87023 CF1PS6 14570100 IC50 = 180 nM T87023 CY04FE 14570101 IC50 = 300 nM T87023 C60WKO 14570103 IC50 = 5 nM T87023 CS0GI2 14570105 IC50 = 4 nM T87023 CG1K0Y 14570107 IC50 = 80 nM T87023 C9LBQ5 14570109 IC50 = 50 nM T87023 CBQ8U2 14570110 IC50 = 18 nM T87023 CX7T3E 14570112 IC50 = 4 nM T87023 CXV8Y9 14570113 IC50 = 140 nM T87023 CWBL85 14570115 IC50 = 60 nM T87023 CDF97J 14850516 IC50 = 180 nM T87023 CWZ3A8 14850517 IC50 = 450 nM T87023 CRT39C 14851835 IC50 = 1000 nM T87023 CK5XD2 14851836 IC50 = 10 nM T87023 CB6XP5 14851837 IC50 = 20 nM T87023 CWIS18 14851839 IC50 = 15 nM T87023 CM41GE 14851844 IC50 = 7 nM T87023 C80GHF 14851845 IC50 = 5 nM T87023 C0NHS1 14851856 IC50 = 130 nM T87023 C10FKJ 14851858 IC50 = 12 nM T87023 C5GWX4 14851859 IC50 = 7 nM T87023 CN7VY9 14851860 IC50 = 5 nM T87023 CA69BW 14851861 IC50 = 3 nM T87023 CF0Z2B 14851862 IC50 = 5 nM T87023 CA92DN 14851865 IC50 = 1 nM T87023 C5DV4H 14851868 IC50 = 45 nM T87023 CZ81OA 14851869 IC50 = 0.7 nM T87023 C81FOY 14851873 IC50 = 2 nM T87023 CJ3KB7 14851874 IC50 = 0.2 nM T87023 CDYS82 14851875 IC50 = 4 nM T87023 CP9L5Z 14851876 IC50 = 0.3 nM T87023 C3T8YL 14851877 IC50 = 0.7 nM T87023 CPO42E 14851878 IC50 = 120 nM T87023 CCV61H 14851879 IC50 = 51 nM T87023 CQW1B5 14851880 IC50 = 12 nM T87023 CM5FR9 14851881 IC50 = 3 nM T87023 CSM85K 14851882 IC50 = 0.6 nM T87023 C5ZI8V 14851883 IC50 = 6 nM T87023 CPT9F1 14851884 IC50 = 5 nM T87023 CAO63B 14851885 IC50 = 4 nM T87023 CMVR73 14851886 IC50 = 1 nM T87023 C74AFK 14851887 IC50 = 1 nM T87023 CX5B6D 14851888 IC50 = 9 nM T87023 CW8KJ0 14851889 IC50 = 5 nM T87023 C1SD9F 14851890 IC50 = 4 nM T87023 CER80G 14851891 IC50 = 7 nM T87023 C5OIB1 14851892 IC50 = 25 nM T87023 CI9AY1 14851893 IC50 = 30 nM T87023 CX8VB1 14851894 IC50 = 1000 nM T87023 C1Q2RE 14851895 IC50 = 100 nM T87023 C35WNI 14851899 IC50 = 20 nM T87023 CB9M3Y 14851902 IC50 = 10 nM T87023 CJLV95 14851905 IC50 = 250 nM T87023 CA0Q3B 14851906 IC50 = 100 nM T87023 CE5Z1I 14851908 IC50 = 5 nM T87023 C05JIQ 14851911 IC50 = 6 nM T87023 CF64SL 14851914 IC50 = 120 nM T87023 CLS4D8 14851915 IC50 = 25 nM T87023 CM4K6U 14851920 IC50 = 200 nM T87023 C7G0EH 14851921 IC50 = 50 nM T87023 C9SRW7 14851922 IC50 = 100 nM T87023 CO0ZI9 14851924 IC50 = 370 nM T87023 C16ELU 14851927 IC50 = 1000 nM T87023 CWBF08 14851929 IC50 = 250 nM T87023 CAXE30 14851930 IC50 = 150 nM T87023 C7XCS6 14851932 IC50 = 100 nM T87023 CT69LI 14885626 IC50 > 50000 nM T87023 C6U7LN 14885627 IC50 = 3400 nM T87023 C0NO3P 14885628 IC50 = 670 nM T87023 C63PKH 14885629 IC50 = 820 nM T87023 CPY89T 14885630 IC50 = 810 nM T87023 C14UWI 14885631 IC50 = 1000 nM T87023 CF7P1W 14885632 IC50 = 3400 nM T87023 CIW2T8 14885633 IC50 = 8700 nM T87023 CR29QH 14885639 IC50 > 50000 nM T87023 C0RCP6 14885640 IC50 > 50000 nM T87023 CAN9H8 14885641 IC50 = 41000 nM T87023 C5Q1FS 14885642 IC50 = 28000 nM T87023 C3N4SC 14894667 IC50 = 1000 nM T87023 CD80TK 14894668 IC50 = 20 nM T87023 CPZD47 14894754 IC50 = 300 nM T87023 CGME82 14894759 IC50 = 500 nM T87023 CIZ82M 14964714 IC50 = 220 nM T87023 CI45CF 14964715 IC50 = 60 nM T87023 CD09PT 14964717 IC50 = 40 nM T87023 C4HNX6 14964719 IC50 = 500 nM T87023 C9E6AV 14964722 IC50 = 50 nM T87023 C25DYC 14964723 IC50 = 89000 nM T87023 C0A2RM 14964724 IC50 = 35000 nM T87023 C7LI9U 14964727 IC50 = 9500 nM T87023 CSH90Y 14964730 IC50 = 1140 nM T87023 CTC74B 15084135 IC50 = 180 nM T87023 CEOH63 15084136 IC50 = 260 nM T87023 CN37TK 15084138 IC50 = 1000 nM T87023 C8O6WV 15084139 IC50 = 1000 nM T87023 CM4F8C 15084140 IC50 = 650 nM T87023 C3E2IX 15084147 IC50 = 100 nM T87023 C3KZ4F 15084148 IC50 = 300 nM T87023 CMW42Z 15084149 IC50 = 380 nM T87023 CMEQ63 15084150 IC50 = 420 nM T87023 C84THB 15084151 IC50 = 400 nM T87023 CZ87IM 15084152 IC50 = 60 nM T87023 C0Q7MH 15084157 IC50 = 35 nM T87023 C3COK9 15084158 IC50 = 8 nM T87023 CGU71E 15084159 IC50 = 20 nM T87023 C57BCL 15084160 IC50 = 20 nM T87023 CT2PW7 15084161 IC50 = 400 nM T87023 CG0PF5 15097565 IC50 = 550 nM T87023 CT87IS 18639456 IC50 = 3 nM T87023 CFG06W 18755202 Ki = 59 nM T87023 C76OSJ 21276953 IC50 = 7.5 nM T87023 C7FP9U 21577212 IC50 = 575.44 nM T87023 CO2T4K 22840724 IC50 > 1000 nM T87023 CJPG51 23214200 IC50 = 278 nM T87023 CQ9XE5 23214230 IC50 = 8 nM T87023 C1GMB3 23214264 IC50 = 33 nM T87023 CYDT52 23214297 IC50 = 585 nM T87023 C0WAM4 23685642 Ki = 110 nM T87023 CI67HD 44273122 IC50 = 75 nM T87023 C9SR4G 44273257 IC50 = 12 nM T87023 C1DAB0 44273266 IC50 = 110 nM T87023 C43OBW 44273268 IC50 = 75 nM T87023 C5Y2XS 44273289 IC50 = 150 nM T87023 CP2GT8 44273297 IC50 = 1000 nM T87023 CYN67I 44273305 IC50 = 6 nM T87023 CM3QV5 44273306 IC50 = 6 nM T87023 CXP37E 44273330 IC50 = 30 nM T87023 CO80DX 44273370 IC50 = 560 nM T87023 C85BUC 44273372 IC50 = 360 nM T87023 C74DMO 44273385 IC50 = 15 nM T87023 CJ6XK2 44273427 IC50 = 90 nM T87023 C6D9OR 44273429 IC50 = 4 nM T87023 C4HD8F 44273438 IC50 = 1000 nM T87023 C4GT8A 44273441 IC50 = 15 nM T87023 CC5Y8H 44273467 IC50 = 25 nM T87023 C2QUX4 44273471 IC50 = 7 nM T87023 CGY7N4 44273479 IC50 = 9 nM T87023 CIO5G9 44273765 IC50 = 70 nM T87023 CCN9H2 44281321 IC50 = 80 nM T87023 C4UJ8B 44281337 IC50 = 10 nM T87023 C83YMH 44281548 IC50 = 110 nM T87023 CX71ET 44281549 IC50 = 120 nM T87023 C9Q7DM 44281731 IC50 = 400 nM T87023 C3Z6QM 44283756 IC50 = 3000 nM T87023 CFC8S1 44283766 IC50 = 4000 nM T87023 CK8J9F 44283767 IC50 = 800 nM T87023 C2UF8A 44283768 IC50 = 5000 nM T87023 CS21BL 44283769 IC50 = 1000 nM T87023 CT5I4V 44283777 IC50 = 18000 nM T87023 CNM40C 44283798 IC50 = 1500 nM T87023 C1OI4A 44283802 IC50 = 100 nM T87023 CLR84V 44283822 IC50 = 2500 nM T87023 CF31SK 44283845 IC50 = 4000 nM T87023 C76TSH 44283848 IC50 = 300 nM T87023 CUZ37Y 44283860 IC50 = 25000 nM T87023 C8JX7R 44283865 IC50 = 150 nM T87023 CZ3XQ8 44283867 IC50 = 6000 nM T87023 CE5D7C 44283890 IC50 = 6000 nM T87023 CF1MN7 44283916 IC50 = 3000 nM T87023 CBE14Q 44283931 IC50 = 1000 nM T87023 C78FQC 44283979 IC50 = 200 nM T87023 C4A3WY 44283998 IC50 = 300 nM T87023 CZ2TY4 44284056 IC50 = 1600 nM T87023 CM7GJ9 44284128 IC50 = 230 nM T87023 CRX4K3 44284129 IC50 = 4000 nM T87023 C7UWD8 44284130 IC50 = 2000 nM T87023 CZB4F1 44284141 IC50 = 4000 nM T87023 C1K3GO 44284155 IC50 = 900 nM T87023 CT2BU0 44284169 IC50 = 15000 nM T87023 C4BQJ8 44284228 IC50 = 500 nM T87023 CTCG71 44284380 IC50 = 190 nM T87023 CH7ZD3 44284397 IC50 = 250 nM T87023 CGYC29 44284425 IC50 = 500 nM T87023 C2OGK8 44284466 IC50 = 300 nM T87023 C06QAE 44284467 IC50 = 100 nM T87023 CA0PI2 44284483 IC50 = 2000 nM T87023 C7ETA6 44284532 IC50 = 3 nM T87023 C6WUT9 44284535 IC50 = 20 nM T87023 CTR6U3 44284549 IC50 = 5 nM T87023 C5M0GN 44284550 IC50 = 10 nM T87023 CEJ54R 44284551 IC50 = 7 nM T87023 C3HV9K 44284580 IC50 = 25 nM T87023 CHKR42 44284581 IC50 = 7 nM T87023 CXBZ65 44284614 IC50 = 15 nM T87023 C5FDO0 44296798 IC50 = 700 nM T87023 C35VIC 44296856 IC50 = 2100 nM T87023 C5VEM4 44297137 IC50 = 55 nM T87023 C7LYV3 44297357 IC50 = 800 nM T87023 C52KZM 44297376 IC50 = 60 nM T87023 CA3F7B 44297384 IC50 > 1000 nM T87023 CF5PW4 44297401 IC50 > 1000 nM T87023 CUN0H2 44297792 Ki = 1 nM T87023 CSNO71 44299770 IC50 = 180 nM T87023 C2E0LD 44328857 IC50 = 30 nM T87023 CC18PX 44328858 IC50 = 7 nM T87023 C01ILU 44328877 IC50 = 40 nM T87023 CA5IU4 44328916 IC50 = 6 nM T87023 C5P1MF 44328930 IC50 = 15 nM T87023 C0DXY1 44329180 IC50 = 26 nM T87023 CFVO05 44329213 IC50 = 33 nM T87023 CP4N1I 44329214 IC50 = 24 nM T87023 C3D6WM 44329219 IC50 = 90 nM T87023 C6PN0F 44329225 IC50 = 55 nM T87023 C1AFG6 44340797 Ki = 1000 nM T87023 C9XFY5 44344131 Ki = 3.72 nM T87023 C1V6ZA 44344325 Ki = 2.86 nM T87023 CLJ8A4 44361141 IC50 > 50000 nM T87023 CXE1H3 44370579 IC50 = 11 nM T87023 C5XWT1 44370606 IC50 = 500 nM T87023 CO2KZ1 44372409 IC50 = 17 nM T87023 C62LFJ 44372410 IC50 = 300 nM T87023 C8T3IA 44372435 IC50 = 1606 nM T87023 C0ZW6D 44372440 IC50 = 17 nM T87023 CG3Y2W 44372459 IC50 = 858 nM T87023 CKS38M 44372461 IC50 = 56 nM T87023 C0N9CI 44372545 IC50 = 26 nM T87023 C8RK3Y 44372629 IC50 = 91 nM T87023 CK4O7N 44372644 IC50 = 68 nM T87023 C4A2EQ 44372678 IC50 = 59 nM T87023 CZ76XE 44386405 IC50 = 100 nM T87023 C21FBR 44399100 IC50 = 1122.02 nM T87023 C4VTG7 44399185 IC50 = 2344.23 nM T87023 CB97LK 44399202 IC50 = 1445.44 nM T87023 CJRG27 54761054 Ki = 2000 nM T87023 C87RWE 71716054 IC50 = 28.9 nM T87023 CAJO25 71716651 IC50 = 58.8 nM T87023 C17KVQ 71720304 IC50 = 40.4 nM T87023 C2YEN3 73356389 IC50 = 1148.15 nM T87023 CPMZ51 135503537 IC50 = 7200 nM T87023 D01CDL 6917920 Ki = 103 nM T87023 D04FHG 108156 Ki = 0.15 nM T87023 D09MAZ 46897162 IC50 > 5000 nM T87023 D0N2WK 107681 IC50 = 600 nM T87023 D0OT3H 132114 IC50 = 12 nM T87023 D0X9RL 9954410 IC50 = 0.015 nM T32764 D0R0MW 5329102 IC50 = 47.4 nM T32764 CHWL84 6539599 IC50 = 220 nM T32764 C6P4BO 6539600 IC50 = 1200 nM T32764 COD03X 10156251 IC50 = 4.32 nM T32764 C3VRO9 44557921 IC50 = 5888.44 nM T32764 C67OJG 44588117 Ki = 541 nM T32764 CKA12O 57891796 IC50 = 209 nM T32764 C8NF7Y 59699998 IC50 = 23.6 nM T32764 CZ14IK 91938067 IC50 = 0.07 nM T32764 CDL4P0 118009188 IC50 = 3.3 nM T32764 C38SJA 118419786 IC50 = 0.3 nM T32764 CE7L5R 118419870 IC50 = 1400 nM T32764 CS2VP0 118420021 IC50 = 3 nM T32764 CY6NG3 118429629 IC50 = 0.51 nM T32764 CNO6Z1 118429823 IC50 = 0.32 nM T32764 C7YZ8X 118429852 IC50 = 0.42 nM T32764 CJB69T 118429935 IC50 = 0.23 nM T32764 C4H7SM 118714184 IC50 = 319 nM T32764 CR2W8V 118864359 IC50 = 4 nM T32764 CI91CV 121255756 IC50 = 6 nM T32764 CYBU50 124002327 IC50 = 18000 nM T32764 C48IAY 134530903 IC50 = 0.62 nM T32764 C4YWO9 134812845 Ki = 9.1 nM T32764 CG15PY 134812846 Ki = 53000 nM T32764 CQBF40 135284803 IC50 = 0.2 nM T32764 CO58DJ 135390126 IC50 = 886 nM T32764 C6AZ2R 135435018 IC50 = 280 nM T32764 C9O8CQ 137348448 Ki = 8.3 nM T32764 C63TGO 137349551 Ki = 6.3 nM T32764 C6I5ME 137349552 Ki = 10 nM T32764 C1UYP7 137640287 IC50 = 2800 nM T32764 C6B9RI 137655689 IC50 = 350 nM T32764 C0B7LO 138393295 IC50 = 4.02 nM T32764 CYZ4A6 146121078 IC50 = 18000 nM T32764 CRC8D2 155489850 Ki = 78000 nM T32764 CUC56L 155515968 IC50 = 3500 nM T32764 C3W9MD 155516193 IC50 = 9.27 nM T32764 CU9P1O 155516654 IC50 = 72.1 nM T32764 CO79KW 155517221 IC50 = 108 nM T32764 CG8J5X 155518911 Ki = 32 nM T32764 C5OK4J 155519508 IC50 = 3800 nM T32764 CD92PB 155519881 IC50 = 381 nM T32764 C0EH9S 155520094 IC50 = 161 nM T32764 C6Y3ZR 155520697 IC50 = 800 nM T32764 CR3LG7 155520971 IC50 = 420 nM T32764 C4FLT9 155521757 IC50 = 54 nM T32764 CF92OZ 155523797 IC50 = 149 nM T32764 C8YX3N 155525320 IC50 = 910 nM T32764 C1LH3X 155533332 IC50 = 387 nM T32764 CAN08J 155534113 Ki = 20 nM T32764 CHCE71 155534845 IC50 = 3390 nM T32764 C16JRL 155535406 Ki = 33 nM T32764 CX0V3J 155535984 IC50 = 370 nM T32764 C3XR8O 155536206 Ki = 22 nM T32764 CN9MV3 155536780 IC50 = 184 nM T32764 C6VQA5 155537429 IC50 > 50000 nM T32764 CHQN92 155537739 IC50 = 1100 nM T32764 CA74KV 155537883 IC50 = 398 nM T32764 C4G0DY 155538489 IC50 = 4440 nM T32764 CDB8Q3 155540035 IC50 = 381 nM T32764 C8Q4LF 155540633 IC50 = 18.6 nM T32764 CX68YN 155541385 Ki > 100000 nM T32764 CWU67H 155543077 Ki = 30 nM T32764 CBT5A1 155543338 IC50 = 230 nM T32764 CD8K3O 155543384 Ki = 44 nM T32764 C4CV6S 155544989 IC50 = 462 nM T32764 CL51KX 155546156 IC50 = 2200 nM T32764 CUTW39 155546618 Ki = 8.2 nM T32764 C4E0HB 155546757 Ki = 59 nM T32764 CR45OK 155547135 IC50 = 560 nM T32764 C49UVQ 155547733 Ki = 8.5 nM T32764 CI2J4O 155551330 Ki = 22 nM T32764 CM1WS6 155552596 IC50 > 50000 nM T32764 CP2K8O 155554487 Ki = 12 nM T32764 CYC93Q 155556093 IC50 = 612 nM T32764 CS8MC1 155562025 Ki = 39 nM T32764 C8UW4P 155562878 Ki = 6.2 nM T32764 CS7TO0 155566480 IC50 = 120 nM T32764 C53HDP 155568011 IC50 = 71 nM T32764 CMHX39 155568223 IC50 = 7700 nM T32764 CDP94M 155569521 Ki = 24 nM T47081 D02EEJ 6479267 Ki = 1.84 nM T47081 D0CE0O 11513676 Ki = 0.34 nM T47081 D0G7UX 5284373 Ki = 2.64 nM T47081 D0M2OY 53259809 Ki = 16800 nM T47081 D08MYL 6473876 Ki = 2.11 nM T47081 CY0Q4V 444384 IC50 = 2000000 nM T47081 CLYE08 497073 IC50 = 6000 nM T47081 C8SG7U 497075 IC50 > 10000000 nM T47081 CAWY91 497076 IC50 = 90000 nM T47081 CC9D3J 497077 IC50 > 10000000 nM T47081 CBMF04 497078 IC50 = 500000 nM T47081 C6KF5Y 1367020 IC50 = 580 nM T47081 CP61UY 2823177 IC50 = 920 nM T47081 CM6OW0 3190778 IC50 = 5.5 nM T47081 CDPT84 4128827 IC50 = 316 nM T47081 C7T6VH 4401642 IC50 = 14 nM T47081 CSQP36 5020377 IC50 = 303 nM T47081 CZ34OX 5116189 IC50 = 5500 nM T47081 C7DIT9 5493631 IC50 = 680000 nM T47081 C35VSF 5493632 IC50 = 1000000 nM T47081 CGN50H 5493634 IC50 = 260000 nM T47081 C8U3AT 5493635 IC50 = 115000 nM T47081 C5I2UC 5493638 IC50 = 280000 nM T47081 CNIC61 6475296 IC50 = 310 nM T47081 C8RA6C 6476061 IC50 = 11.1 nM T47081 CTXB32 6479257 IC50 = 3 nM T47081 CMH26D 6479258 IC50 = 47 nM T47081 C45EVU 6479259 IC50 = 15 nM T47081 CQ1X3C 6479260 IC50 = 61 nM T47081 C1YMW4 6479261 IC50 = 277 nM T47081 CAYZ53 6479262 IC50 = 97 nM T47081 CPCG74 6479263 IC50 = 128 nM T47081 C16CZK 6479264 IC50 = 19 nM T47081 CN1BF8 6479265 IC50 = 165 nM T47081 C8N4YK 6479266 IC50 = 110 nM T47081 CAGX82 6479268 IC50 = 6047 nM T47081 CM36KU 6479269 IC50 = 1572 nM T47081 CJWU53 6479270 IC50 = 882 nM T47081 CRV94O 6479271 IC50 = 959 nM T47081 C03LTJ 10034324 IC50 = 934 nM T47081 CODJ10 10626583 Ki = 795 nM T47081 CO9XA6 10819131 IC50 = 1500000 nM T47081 CF45ID 11516665 IC50 = 20 nM T47081 CGP87C 11531251 IC50 = 951 nM T47081 CSY31B 11559871 IC50 = 748 nM T47081 C6M1ZU 11567780 IC50 = 320 nM T47081 CJ27OG 11588606 IC50 = 140 nM T47081 CN8M2B 11617502 IC50 = 71 nM T47081 CS2Y6M 11631957 IC50 = 60 nM T47081 CX63ZC 11632684 IC50 = 60 nM T47081 CLP34W 11638938 IC50 = 592 nM T47081 CS3YJ8 11660364 IC50 = 640 nM T47081 C37WLM 11675245 IC50 = 528 nM T47081 C3SK8D 11703833 IC50 = 880 nM T47081 C2QN6F 11710570 IC50 = 1437 nM T47081 C73OMC 11717355 IC50 = 458 nM T47081 C89EKB 11718015 IC50 = 499 nM T47081 CUY92Q 13422114 IC50 = 130 nM T47081 CC6XY7 13578707 IC50 = 350 nM T47081 C8KA7W 20415061 IC50 = 460 nM T47081 C31GDL 24814873 IC50 = 14 nM T47081 C2ON4L 25044910 IC50 = 690 nM T47081 CY8HB6 25046022 IC50 = 330 nM T47081 CT2E3I 25098032 IC50 = 590 nM T47081 CK0P2Q 42630203 IC50 = 650 nM T47081 C69CNK 44248910 IC50 > 10000 nM T47081 C46XEC 44248911 IC50 = 103 nM T47081 CS6N9K 44248912 IC50 = 71.2 nM T47081 CHX9S4 44248913 IC50 = 159 nM T47081 CSDG42 44248914 IC50 > 10000 nM T47081 CJT1A8 44249039 IC50 = 364 nM T47081 CVW1T9 44249040 IC50 = 263 nM T47081 CNFI87 44249041 IC50 = 2.59 nM T47081 CW6LT7 44249042 IC50 = 1.52 nM T47081 C7U6PN 44249044 IC50 = 1910 nM T47081 C1HPV8 44249170 IC50 > 10000 nM T47081 CW4AU3 44249173 IC50 = 12.1 nM T47081 CKO3I0 44249174 IC50 > 10000 nM T47081 CL7M2J 44249303 IC50 = 620 nM T47081 C97JUQ 44249304 IC50 > 10000 nM T47081 C0SVJ1 44249305 IC50 = 31.6 nM T47081 CA3K2N 44249306 IC50 > 10000 nM T47081 CBEL85 44249307 IC50 = 370 nM T47081 C5M4VW 44249309 IC50 = 136 nM T47081 CR2K7N 44249310 IC50 > 10000 nM T47081 C57MCG 44249414 IC50 > 10000 nM T47081 CSJD94 44249415 IC50 > 10000 nM T47081 CER54N 44294512 IC50 = 2500000 nM T47081 CKYA61 44294584 IC50 = 850000 nM T47081 C4R1DL 44294708 IC50 > 10000000 nM T47081 CTE19D 44294709 IC50 > 10000000 nM T47081 CT5IJ4 44294814 IC50 = 2800000 nM T47081 C4GLS0 44294838 IC50 = 760000 nM T47081 C5EQ7U 44295020 IC50 = 1300000 nM T47081 CHI01J 44295050 IC50 = 1500000 nM T47081 CS5I9W 44295136 IC50 = 970000 nM T47081 COCG50 44295258 IC50 = 820000 nM T47081 CV7PD8 44341483 IC50 = 48 nM T47081 C5M1FB 44341507 IC50 = 256 nM T47081 CM9L8P 44365970 IC50 = 1500000 nM T47081 C50FPJ 44366040 IC50 = 2500000 nM T47081 C0JKL6 44366208 IC50 = 2600000 nM T47081 C98VGM 44366209 IC50 = 165000 nM T47081 C6PCZ9 44366232 IC50 = 850000 nM T47081 CRES48 44366233 IC50 = 325000 nM T47081 C7AQ3R 44366260 IC50 = 2100000 nM T47081 CS74HY 44366261 IC50 = 970000 nM T47081 CEH4W6 44366303 IC50 = 820000 nM T47081 CF3B2I 44366350 IC50 = 260000 nM T47081 C0I3BR 44366351 IC50 = 760000 nM T47081 C9HQ5S 44366390 IC50 = 2800000 nM T47081 CY89LF 44366391 IC50 = 1300000 nM T47081 CDJ21S 44366404 IC50 = 500000 nM T47081 CPW1A7 44366405 IC50 = 90000 nM T47081 C4SQ1N 44366450 IC50 = 280000 nM T47081 CUI2X6 44366451 IC50 = 6000 nM T47081 CMCP73 44366452 IC50 = 365000 nM T47081 C2LG1F 44366453 IC50 = 115000 nM T47081 C5Q4VN 44393426 Ki = 100 nM T47081 CP57YU 44393427 Ki = 75 nM T47081 CGX7M4 44393512 Ki = 10 nM T47081 CGP76Z 44393513 Ki = 24 nM T47081 CU0RC4 44393514 Ki = 18 nM T47081 CZAD42 44406917 IC50 = 4100 nM T47081 C0FLH5 44582698 IC50 = 740 nM T47081 C0ON5I 44582699 IC50 = 810 nM T47081 CW3R7N 44582757 IC50 = 740 nM T47081 CCV89D 44582780 IC50 = 880 nM T47081 CZM71K 44582804 IC50 = 600 nM T47081 CWF96D 44582805 IC50 = 450 nM T47081 CYN7C5 44582823 IC50 = 160 nM T47081 CW4P8K 44582824 IC50 = 450 nM T47081 CX94NI 45138814 IC50 = 2.4 nM T47081 CN72XD 45269870 IC50 > 10000 nM T47081 CS30FH 49863381 IC50 = 206 nM T47081 C3YI2V 49863382 IC50 = 950 nM T47081 CS48JU 49863383 IC50 = 4.75 nM T47081 CWI47U 50899161 IC50 = 26.6 nM T47081 CHN71J 52940634 IC50 = 31.2 nM T47081 CQ83LE 52940669 IC50 = 22.9 nM T47081 C2H0IK 52940670 IC50 = 46 nM T47081 CPKZ45 52940671 IC50 = 35.2 nM T47081 C7MA9P 52941831 IC50 = 9.12 nM T47081 CH9QA8 52941859 IC50 = 21.4 nM T47081 C97YWD 52945243 IC50 = 26.7 nM T47081 CE05IO 52945473 IC50 = 218 nM T47081 C43LWJ 52945496 IC50 = 140 nM T47081 C3BCG7 52946681 IC50 = 83.5 nM T47081 CR63JF 52946682 IC50 = 22.8 nM T47081 CH8TZ9 52946683 IC50 = 103 nM T47081 C7KW3U 52947912 IC50 = 23 nM T47081 C4KAU1 52947949 IC50 = 662 nM T47081 CGX04A 52947950 IC50 = 65.2 nM T47081 CS90AU 52952820 IC50 = 33.11 nM T47081 CBWK59 53321090 Ki = 106 nM T47081 CNS79R 53344622 IC50 = 2.7 nM T47081 CPD19A 53357115 IC50 = 350 nM T47081 CMYW90 53357116 IC50 = 630 nM T47081 C75LWY 53357117 IC50 = 500 nM T47081 C40GVQ 53357247 IC50 = 360 nM T47081 CC0Y1S 53357248 IC50 = 390 nM T47081 CPM2F7 53357386 IC50 = 330 nM T47081 COP18F 53357507 IC50 = 520 nM T47081 C4P3GC 53357508 IC50 = 420 nM T47081 C4O0YX 53357509 IC50 = 4.1 nM T47081 C96CAE 53357630 IC50 = 450 nM T47081 C8C9ZH 53358962 IC50 = 1.1 nM T47081 C3VJ0N 56668120 IC50 = 2000000 nM T47081 C30PVF 56675024 IC50 = 2600000 nM T47081 CFMP72 56678333 IC50 = 2100000 nM T47081 CFAY29 56678334 IC50 = 165000 nM T47081 CQB1I0 57384849 Ki = 14 nM T47081 CZK8P2 57384850 Ki = 65 nM T47081 CX67HU 57385085 Ki = 4 nM T47081 C6PXU0 57398046 IC50 = 4.9 nM T47081 C6ZK4A 67978739 Ki = 16 nM T47081 C6RT1L 71590783 IC50 = 740 nM T47081 CC0TY2 71590784 IC50 = 810 nM T47081 CH23LT 71596756 IC50 = 550 nM T47081 CZOT97 71596824 IC50 = 380 nM T47081 CC37ZO 71596825 IC50 = 330 nM T47081 C2IJ6X 71596826 IC50 = 460 nM T47081 CSE28O 73333514 Ki = 23 nM T47081 CDF54U 73333515 Ki = 10.7 nM T47081 CKS08Z 73333613 Ki = 12.4 nM T47081 C5FWY3 73333614 Ki = 43.9 nM T47081 C2LR7I 73333729 Ki = 11.8 nM T47081 CQH16I 73333730 Ki = 36.6 nM T47081 CRA39X 73333846 Ki = 57.7 nM T47081 C47PVY 73347049 IC50 = 680000 nM T47081 CKV1A9 73348786 IC50 = 2.3 nM T47081 CIXM26 73353051 IC50 = 16 nM T47081 C5J6GK 122437357 IC50 = 11.2 nM T47081 CUKL46 127038149 IC50 = 10000 nM T47081 CF7KS5 127038150 IC50 = 10000 nM T47081 C6HPE3 127038151 IC50 = 10000 nM T47081 CQC1L7 127038489 IC50 = 940 nM T47081 CI8EO6 127039060 IC50 = 10000 nM T47081 C7NW5Q 127039075 IC50 = 2760 nM T47081 CSU85H 127039831 IC50 = 10430 nM T47081 CA1P8V 127039832 IC50 = 10260 nM T47081 C2JQ4V 127039851 IC50 = 10000 nM T47081 C1DTR2 127039852 IC50 = 1220 nM T47081 CI03BD 127040172 IC50 = 10800 nM T47081 C0OTQ9 127040173 IC50 = 10000 nM T47081 CA75UB 127040174 IC50 = 10000 nM T47081 CC0GN1 127040175 IC50 = 10000 nM T47081 C8PI2G 127041686 IC50 = 10000 nM T47081 CS0EM4 127041788 IC50 = 10330 nM T47081 CE0KL8 127041789 IC50 = 10000 nM T47081 C35DGM 127042320 IC50 = 11620 nM T47081 C2VGI1 136220121 Ki = 64.7 nM T47081 C2ZA8L 137348679 Ki = 7 nM T47081 CY46VP 137637353 Ki = 4.3 nM T47081 D04PGW 6475368 IC50 = 166 nM T47081 D07ABJ 44358392 IC50 = 783 nM T47081 D07IQR 11639129 IC50 = 361 nM T47081 D0P6TX 3663276 IC50 = 754 nM T47081 D0X5JR 11574097 IC50 = 810 nM T22583 D01TNW 9887712 IC50 = 1.35 nM T22583 D0Q3VE 44814423 IC50 = 0.877 nM T22583 CQW18C 10133993 IC50 = 42 nM T22583 C0H4YI 11509368 IC50 = 19 nM T22583 C67HDU 11516541 IC50 = 11 nM T22583 CGY18M 11517178 IC50 = 120 nM T22583 CKI73F 11530288 IC50 = 690 nM T22583 CXD1G4 11531141 IC50 = 120 nM T22583 CH01CX 11552436 IC50 = 29 nM T22583 CTR8Z2 11560149 IC50 = 110 nM T22583 C3I5OZ 11631863 IC50 = 290 nM T22583 C0U9BG 11639042 IC50 = 59 nM T22583 C4D1CR 11660874 IC50 = 150 nM T22583 CW54RB 11675148 IC50 = 28 nM T22583 CFAP86 11682042 IC50 = 630 nM T22583 CQM7K2 11718002 IC50 = 150 nM T22583 C87XZS 46206829 IC50 = 6.98 nM T22583 CNI2X3 52952611 IC50 = 43.1 nM T22583 CK7EW5 52952725 IC50 = 0.882 nM T22583 CH03OA 52952726 IC50 = 89.9 nM T22583 C7A5FM 54580749 IC50 = 1.07 nM T22583 C05HIX 54580768 IC50 = 103 nM T22583 CH90AV 54580792 IC50 = 81.9 nM T22583 C9LET3 54582741 IC50 = 89.6 nM T22583 C57FRI 54582776 IC50 = 99.7 nM T22583 CP3HT2 54583734 IC50 = 59.5 nM T22583 CW6H2Y 54586611 IC50 = 1.11 nM T22583 D03AJS 10177526 IC50 = 4.8 nM T22583 D06WAL 6072 IC50 = 16 nM T22583 D0X1TN 9824918 IC50 = 260 nM T96623 D01BYB 5957 IC50 = 893677 nM T96623 D08IBS 190 IC50 > 4000000 nM T96623 D0Q0PR 54675769 IC50 = 231000 nM T96623 D01FYA 9549213 EC50 = 10.2 nM T96623 D02PGP 448965 EC50 = 15000 nM T96623 D02TTL 44156921 IC50 = 38 nM T96623 D05BYA 135539077 Ki = 0.064 nM T96623 D05HWN 16736529 Ki = 1.7 nM T96623 D06YSP 11955716 IC50 = 350 nM T96623 D09XGB 135446210 IC50 = 28 nM T96623 D0F3NF 67501411 Ki = 21.3 nM T96623 D0I1QI 135564985 IC50 = 5 nM T96623 D0U2BH 65064 IC50 = 155000 nM T96623 D03BNU 59604787 IC50 > 3500 nM T96623 CES15Y 6942 IC50 > 4000000 nM T96623 COUI64 79856 IC50 = 570000 nM T96623 CXI2U0 156194 IC50 = 110000 nM T96623 CDZ65K 199472 IC50 = 34000 nM T96623 C2GU6I 214051 IC50 = 350000 nM T96623 CA23LP 448972 IC50 = 660 nM T96623 CN2TZ3 579787 IC50 = 490000 nM T96623 CJUN-71 658498 IC50 = 9000 nM T96623 CIV7A0 745543 IC50 > 50000 nM T96623 C3U5ZX 893376 Ki = 32200 nM T96623 C4GB8N 1367558 IC50 = 700 nM T96623 CR69HB 1916699 IC50 = 900 nM T96623 C6KN2W 3695754 IC50 = 1560 nM T96623 CQCH29 5287469 IC50 = 258 nM T96623 C4ODB9 5287470 IC50 = 461 nM T96623 C3UB9I 6478909 IC50 = 90 nM T96623 CODT42 6914564 EC50 = 38.8 nM T96623 C3RL9A 9844790 IC50 = 30000 nM T96623 CGDO38 9887768 IC50 = 24000 nM T96623 CA0I2C 9931416 IC50 = 64000 nM T96623 CU9SK6 10183346 IC50 = 280 nM T96623 CYQP95 11198704 IC50 > 100000 nM T96623 CO3F6K 11221466 IC50 > 100000 nM T96623 CH4B2Z 11223683 IC50 > 200000 nM T96623 CNA8U5 11290334 IC50 = 340 nM T96623 CBZS48 11302159 IC50 > 300000 nM T96623 CDJX31 11326407 IC50 > 100000 nM T96623 C2ZCY3 11336657 IC50 > 300000 nM T96623 CIRH67 11349446 IC50 > 300000 nM T96623 CUO6Q7 11393625 IC50 > 100000 nM T96623 CZ05EG 11405422 IC50 = 80 nM T96623 CXN76P 11406285 IC50 > 500000 nM T96623 CP3Z4O 11407267 IC50 > 100000 nM T96623 CZKO68 11407809 EC50 = 30 nM T96623 C40WGT 11415286 IC50 = 5700 nM T96623 CR9IQ7 11450570 IC50 > 300000 nM T96623 C8VZQ6 11463506 IC50 > 100000 nM T96623 CI53RD 11473241 IC50 > 100000 nM T96623 CK4VD6 11484509 IC50 = 300 nM T96623 C84KRP 11512802 IC50 = 90 nM T96623 CJGE43 11519125 IC50 = 14 nM T96623 C05VSM 11539274 EC50 = 30.5 nM T96623 CNJ5W1 11562562 EC50 = 22 nM T96623 CG83HO 11568559 EC50 > 15000 nM T96623 CS96GN 11598450 EC50 > 15000 nM T96623 CEW1A8 11627094 EC50 = 22.3 nM T96623 C24EXR 11661053 EC50 = 51.2 nM T96623 CUY74F 11677337 EC50 = 10.8 nM T96623 CKYR08 11704110 EC50 = 4500 nM T96623 C79VTC 11773074 IC50 > 50000 nM T96623 C9X1CE 11835438 IC50 = 5310 nM T96623 C38WXA 11849869 IC50 = 110 nM T96623 CS89EP 11850701 IC50 = 28 nM T96623 CU0PD4 11850702 IC50 = 30 nM T96623 CZ8OW4 11850766 IC50 = 110 nM T96623 C0QP7W 11850832 IC50 = 180 nM T96623 CIP75F 11850896 IC50 = 30 nM T96623 C5QF7K 11855741 IC50 = 47 nM T96623 C5LYR8 11856019 IC50 = 176 nM T96623 CO6S8Z 11978672 IC50 = 1300 nM T96623 C7MVC0 11978794 IC50 = 900 nM T96623 CE8M7K 12318923 IC50 = 20000 nM T96623 C30TAB 16028137 IC50 = 63200 nM T96623 CRU65D 16028167 IC50 = 74680 nM T96623 C67IRF 16067745 Ki = 24500 nM T96623 CJ5S6H 16067841 Ki = 12800 nM T96623 C0BQ1Z 16067845 Ki = 661 nM T96623 CAXK01 16210774 IC50 = 80760 nM T96623 CCYS46 16735061 IC50 = 20 nM T96623 CA27TO 16738716 Ki = 195 nM T96623 C84JYD 17755583 Ki = 4000 nM T96623 C5GDL4 20960605 IC50 > 100000 nM T96623 CK7V0T 20960630 IC50 = 55120 nM T96623 C1NF2X 20960632 IC50 = 50900 nM T96623 CV1P0F 20960773 IC50 = 87960 nM T96623 CL7UB4 20960831 IC50 = 59280 nM T96623 CYUK19 20960908 IC50 = 46130 nM T96623 C74FSV 20960914 IC50 = 35180 nM T96623 CUWD49 20960921 IC50 = 47880 nM T96623 CI1M4N 20960922 IC50 = 40240 nM T96623 CO1J8T 21781998 IC50 = 1250000 nM T96623 CX64PD 24875481 Ki = 204 nM T96623 CJMR47 24875482 Ki = 358 nM T96623 C76JLK 24875483 Ki > 200000 nM T96623 C35LJH 24875570 Ki > 200000 nM T96623 CL2HD3 24875573 Ki = 2830 nM T96623 CZ1XL8 24875574 Ki = 2640 nM T96623 C9XLB1 24875575 Ki > 50000 nM T96623 CZJP07 24875576 Ki = 628 nM T96623 CYXD12 24875663 Ki = 4070 nM T96623 C02APU 24875664 Ki = 1720 nM T96623 CA18VT 24875749 Ki < 1 nM T96623 CSAO83 24875750 Ki = 62 nM T96623 CGI85O 24875752 Ki = 4 nM T96623 CT4EZ5 24875845 Ki = 2 nM T96623 CLHP80 24875846 Ki = 8 nM T96623 CN8E5O 24875848 Ki = 7 nM T96623 CS0K2J 24875942 Ki < 1 nM T96623 C9SJO6 24876030 Ki > 200000 nM T96623 CCK0R3 24876378 Ki = 3 nM T96623 C1D5UA 24876379 Ki = 12 nM T96623 CDV0W8 24876453 Ki = 172 nM T96623 COP50W 25060727 IC50 = 731 nM T96623 C2ZP1O 25060728 IC50 = 1898 nM T96623 C5N2MH 25060729 IC50 = 665 nM T96623 CAUB14 25060984 IC50 = 16960 nM T96623 CAU90R 25061236 IC50 > 20000 nM T96623 CI2Z9X 25061495 IC50 = 705 nM T96623 CK7HA1 25061752 IC50 = 4 nM T96623 CHY40D 25061755 IC50 = 7369 nM T96623 C05ACR 25061756 IC50 = 401 nM T96623 CMK7L5 25061757 IC50 = 7752 nM T96623 C1FM3V 25062295 IC50 > 20000 nM T96623 CW52AT 25062560 IC50 > 20000 nM T96623 C9B8GU 25062565 IC50 = 4510 nM T96623 CDZ90V 25062832 IC50 = 5813 nM T96623 C16AFP 25063092 IC50 = 9974 nM T96623 CXMF62 25063093 IC50 = 498 nM T96623 C6OJM4 25063096 IC50 = 3783 nM T96623 CD85QK 25210273 IC50 = 58 nM T96623 CMGK93 25210274 IC50 = 127 nM T96623 CK0AM3 25216601 Ki < 1 nM T96623 C3PZ7E 25216602 Ki < 1 nM T96623 CO96HG 25216724 Ki < 1 nM T96623 C1OJ3B 25216725 Ki < 1 nM T96623 C1YH7K 25216726 Ki < 1 nM T96623 C6ZBI2 25216727 Ki < 1 nM T96623 C76IDS 25216728 Ki = 3 nM T96623 C58RZL 25216729 Ki < 1 nM T96623 COYP08 25216862 Ki = 2 nM T96623 CZ8Y1F 25216863 Ki < 1 nM T96623 C6W8GD 25216865 Ki < 1 nM T96623 CEI92N 25216866 Ki < 1 nM T96623 CN72XP 25216867 Ki = 2 nM T96623 CD0PL1 25216988 Ki = 5 nM T96623 CY1GB3 25217102 Ki < 1 nM T96623 CU18KT 44129601 IC50 = 230 nM T96623 C7VWX5 44220300 IC50 = 56 nM T96623 C2OUE0 44220301 IC50 = 80 nM T96623 C65TNC 44220303 IC50 = 84 nM T96623 CA27ZC 44220304 IC50 = 535000 nM T96623 C5QK7O 44220504 IC50 = 720 nM T96623 CN5OX3 44220706 IC50 = 64 nM T96623 CRK4H7 44220707 IC50 = 80 nM T96623 C5RVU8 44220708 IC50 = 29 nM T96623 CET63I 44220709 IC50 = 102 nM T96623 C76OZA 44220911 IC50 = 58 nM T96623 C2UWT8 45162180 IC50 = 119500 nM T96623 CTO70M 45267899 IC50 = 87 nM T96623 C2Y6QS 50938552 Ki = 12 nM T96623 CSOD41 51035659 Ki = 56 nM T96623 C6G3WF 51035661 Ki = 179 nM T96623 C9NYP4 51036677 Ki = 81 nM T96623 CM8YT7 51036678 Ki = 88 nM T96623 CE59YM 51036893 Ki = 690 nM T96623 CT9Y4W 51037110 Ki > 10000 nM T96623 C4WRY3 51037112 Ki = 5 nM T96623 C0NIJ3 51037321 Ki = 332 nM T96623 CAG39W 51037322 Ki = 45 nM T96623 CUOH43 51037522 Ki = 79 nM T96623 C28LGR 51037524 Ki = 84 nM T96623 CMS6O0 51037525 Ki = 30 nM T96623 CQK26H 51037526 Ki = 64 nM T96623 CD8YO3 51037732 Ki = 87 nM T96623 CI4Q1U 51037733 Ki = 656 nM T96623 CTR6D4 51037734 Ki > 5000 nM T96623 C92ICH 51037945 Ki = 257 nM T96623 CM9IE8 51037946 Ki > 10000 nM T96623 CRI28Z 51037948 Ki = 9 nM T96623 C2PF6K 51037950 Ki > 5000 nM T96623 CXW86J 51038171 Ki = 34 nM T96623 CXW36H 51038406 Ki > 5000 nM T96623 CF56SO 53389265 IC50 = 30 nM T96623 CJZ5F6 53393801 IC50 > 50000 nM T96623 CJS98I 54697785 IC50 = 15300 nM T96623 C7XDW6 54764514 IC50 = 35000 nM T96623 C1VOE8 56593967 IC50 = 50000 nM T96623 C7L5HJ 57402674 IC50 = 1300 nM T96623 CRPW54 59213785 IC50 = 16840 nM T96623 CFM6S1 59213787 IC50 = 568 nM T96623 CJ7DQ0 59213791 IC50 = 3655 nM T96623 CU10OR 66973803 IC50 > 500000 nM T96623 CDA3Q0 66973853 IC50 > 500000 nM T96623 C1RC6B 66973894 IC50 > 500000 nM T96623 C9J1EK 66973895 IC50 > 500000 nM T96623 CM68JH 67042612 Ki = 3500 nM T96623 C19OXR 67042930 Ki = 2100 nM T96623 CI8SM5 67042932 Ki = 2600 nM T96623 C0KQW2 67043239 Ki = 2400 nM T96623 CV8B0R 67495834 Ki = 4 nM T96623 COU0W3 68106001 Ki = 35 nM T96623 CGWN96 68381039 IC50 > 500000 nM T96623 CP6WN0 69927716 Ki = 8400 nM T96623 C29DGL 69927905 Ki = 3100 nM T96623 CJI9A4 69927927 Ki = 6100 nM T96623 C0C6AV 70688271 IC50 = 900 nM T96623 CA1RF5 70690282 IC50 = 21000 nM T96623 COK1T5 71449572 Ki < 1 nM T96623 CHP17T 71451379 Ki < 1 nM T96623 C08PDT 71453186 Ki = 5230 nM T96623 CRD7F8 71454924 Ki < 1 nM T96623 CLQ38U 71454925 Ki > 200000 nM T96623 CO65GF 71456708 Ki > 200000 nM T96623 CA7PH5 71458551 Ki > 200000 nM T96623 CIG6P3 71660550 IC50 > 500000 nM T96623 C79AGJ 71660551 IC50 = 41800 nM T96623 C3O9JC 71740605 IC50 = 52000 nM T96623 C5JFW8 71740714 IC50 = 7000 nM T96623 CAO6B1 71740715 IC50 = 7000 nM T96623 CUE04B 71740716 IC50 = 7000 nM T96623 CFMY78 71741202 IC50 = 16000 nM T96623 C49WST 72190987 IC50 = 63000 nM T96623 C9CW5M 73437615 Ki = 26 nM T96623 CUD54E 73437616 Ki = 5 nM T96623 C25ERP 76310950 IC50 = 9780 nM T96623 CWJ1L0 76310951 IC50 = 5120 nM T96623 CLJP90 76310952 IC50 = 2430 nM T96623 CP7L2S 76310953 IC50 = 2250 nM T96623 C1K4SV 76310954 IC50 = 2030 nM T96623 CCY6L2 76310955 IC50 = 6420 nM T96623 CVC73S 76314590 IC50 = 3670 nM T96623 CCF79Y 76314772 IC50 > 500000 nM T96623 C2XAR1 76314773 IC50 > 500000 nM T96623 CCH78R 76318163 IC50 = 70430 nM T96623 CX25TF 76318373 IC50 > 500000 nM T96623 C2YW9M 76318374 IC50 > 500000 nM T96623 CUZ24J 76321861 IC50 = 920 nM T96623 CTLE58 76321862 IC50 = 970 nM T96623 C0N8VY 76321863 IC50 = 950 nM T96623 CM7TG6 76321864 IC50 = 8690 nM T96623 CVL72G 76322052 IC50 > 500000 nM T96623 CS0PB2 76324772 Ki = 125 nM T96623 C20ISC 76325492 IC50 = 1210 nM T96623 CN1QK9 76325493 IC50 = 13840 nM T96623 CV3OF8 76325494 IC50 = 30410 nM T96623 C1Z0BW 76325495 IC50 = 25770 nM T96623 CO79DQ 76325496 IC50 = 36490 nM T96623 CSW70U 76325497 IC50 = 6320 nM T96623 CN0PO6 76325498 IC50 = 1430 nM T96623 C64XAH 76325678 IC50 > 500000 nM T96623 CI5EZ4 76329032 IC50 = 4370 nM T96623 C6QC1J 76329033 IC50 = 11450 nM T96623 C4WJF9 76329034 IC50 = 750 nM T96623 CN2V4Q 76329035 IC50 = 11790 nM T96623 CZ5BK3 76329241 IC50 > 250000 nM T96623 C9VMX4 76332714 IC50 = 1030 nM T96623 CXA52Z 76332715 IC50 = 870 nM T96623 CB5QW6 76332716 IC50 = 640 nM T96623 C5H0KA 76336314 IC50 = 21230 nM T96623 C7UIH2 76336315 IC50 = 5430 nM T96623 CPHU63 76336316 IC50 = 22610 nM T96623 CW39IX 76336317 IC50 = 15290 nM T96623 C3TF7W 76336318 IC50 > 100000 nM T96623 CB7CF6 86765150 IC50 = 100 nM T96623 CLPF74 88415340 IC50 = 150000 nM T96623 CJ3Q4H 90654630 Ki = 5 nM T96623 CG8S1L 90654631 Ki = 3 nM T96623 CDIY85 90654632 Ki = 39 nM T96623 CV9YA4 90654633 Ki = 56 nM T96623 CRH14E 90654634 Ki = 140 nM T96623 C26WSJ 90654635 Ki = 120 nM T96623 CXLQ38 90654636 Ki = 15 nM T96623 C9F5UB 90654637 Ki = 10 nM T96623 CZ2MP4 90654638 Ki = 20 nM T96623 C17RWB 90654639 Ki = 40 nM T96623 C7X8WK 90654640 Ki = 31 nM T96623 CJ2ZM3 90654641 Ki = 35 nM T96623 C21FPZ 90654642 Ki = 12 nM T96623 C9ZTU1 90654643 Ki = 19 nM T96623 CTB60Y 90654644 Ki = 60 nM T96623 C81JGB 90654645 Ki = 25 nM T96623 CKM2W0 90654646 Ki = 21 nM T96623 CS8U1X 90654647 Ki = 48 nM T96623 CUE4I6 90654648 Ki = 29 nM T96623 CM5JP8 90654649 Ki = 22 nM T96623 CH8FD0 90654650 Ki = 25 nM T96623 C5DP2C 90654651 Ki = 22 nM T96623 CU87TN 90654652 Ki = 30 nM T96623 C4PJ1V 90654653 Ki > 10000 nM T96623 C2TYR0 90654654 Ki = 590 nM T96623 C6SI7L 90654655 Ki > 10000 nM T96623 CG2JK7 90654656 Ki = 420 nM T96623 CBWT05 90654657 IC50 = 27 nM T96623 C6SK1Z 90654658 Ki = 40 nM T96623 C2TLY1 90654659 Ki > 10000 nM T96623 C3R1DJ 90654660 Ki = 1500 nM T96623 CT1QI5 90654661 Ki > 10000 nM T96623 CU8Q1V 90654662 Ki > 10000 nM T96623 CS42OM 90654663 Ki = 2600 nM T96623 C7M8TA 90654664 Ki = 2900 nM T96623 C1H5WC 90654665 Ki = 580 nM T96623 CQ5C1D 90654949 IC50 = 40360 nM T96623 C2R0AG 90654950 IC50 = 27210 nM T96623 CK9I4Z 90654951 IC50 = 24480 nM T96623 CL3F0Z 90654952 IC50 = 7880 nM T96623 CJ0LK6 90654953 IC50 = 3230 nM T96623 C5ED8U 90654954 IC50 = 930 nM T96623 C0AZ8F 90654955 IC50 = 310 nM T96623 CC2MG9 90656416 IC50 = 41000 nM T96623 CQ9B6T 90656417 IC50 = 58000 nM T96623 CJ98AZ 90656418 IC50 = 75000 nM T96623 CC6R0B 90656419 IC50 = 44000 nM T96623 C6LE1I 90656420 IC50 = 98000 nM T96623 C5U8CT 90656421 IC50 = 280000 nM T96623 CZ21XA 90656422 IC50 = 65000 nM T96623 CWF30N 90656423 IC50 = 81000 nM T96623 C5MUP1 90656424 IC50 = 310000 nM T96623 C4BTE5 90656425 IC50 = 410000 nM T96623 C9G0JH 90656426 IC50 = 120000 nM T96623 CUTV54 117889766 IC50 > 100000 nM T96623 CGM51T 117890044 IC50 > 100000 nM T96623 C37QWO 117890084 IC50 > 100000 nM T96623 C1APC8 117890111 IC50 = 39470 nM T96623 CZ4EN5 117890133 IC50 > 100000 nM T96623 CO2R1E 117890146 IC50 > 100000 nM T96623 CX6V7Q 117890195 IC50 > 100000 nM T96623 CLH49C 117890268 IC50 > 100000 nM T96623 CLHP30 117890308 IC50 > 100000 nM T96623 CO25TC 117890352 IC50 > 100000 nM T96623 CA15DJ 117890354 IC50 > 100000 nM T96623 C3R9DT 117890494 IC50 > 100000 nM T96623 C41OJH 118706055 Ki = 22700 nM T96623 CHJ2Q4 118706056 Ki = 28600 nM T96623 CL46VZ 118706057 Ki = 16700 nM T96623 C0ACG5 118706058 Ki = 23400 nM T96623 CRE19B 118706213 Ki = 15200 nM T96623 CY7BI2 118706214 Ki = 1 nM T96623 CT95MR 118724465 IC50 > 160000 nM T96623 C34GFC 118724470 IC50 = 18600 nM T96623 CH78IS 118724472 IC50 = 18800 nM T96623 CL2DG5 118724473 IC50 = 15800 nM T96623 C2R1GL 118724474 IC50 > 120000 nM T96623 CMT73D 118724475 IC50 > 67000 nM T96623 CFIO82 118724476 IC50 = 121000 nM T96623 CF3Q1W 118724477 IC50 = 10400 nM T96623 CQP10T 118724478 IC50 = 16800 nM T96623 C9NO7P 118724479 IC50 > 27000 nM T96623 C6UBV8 118724480 IC50 = 730 nM T96623 CISE62 135431462 IC50 = 740 nM T96623 CF07JI 135464271 IC50 = 600 nM T96623 CD4H2W 135467994 IC50 = 87000 nM T96623 CBX3Q2 135566391 IC50 = 7600 nM T96623 CWT67P 135566392 IC50 > 50000 nM T96623 CEK31P 135566415 IC50 = 30 nM T96623 CO9SP6 135566717 IC50 = 45000 nM T96623 C3KUM1 135895337 IC50 = 55 nM T96623 CDT3O1 135895338 IC50 = 153 nM T96623 C2I7BL 135895339 IC50 = 74 nM T96623 C6E1DK 135895340 IC50 = 167 nM T96623 C3YCS4 135895341 IC50 = 168 nM T96623 C8BU7Z 135895348 IC50 = 41 nM T96623 CJ64AE 135895349 IC50 = 120 nM T96623 CF7K4Y 135895351 IC50 = 71 nM T96623 CVGA81 135895352 IC50 = 260 nM T96623 C86SWI 135895353 IC50 = 240 nM T96623 C3BH0Q 135895354 IC50 = 30 nM T96623 CZLE25 135895361 IC50 = 40 nM T96623 CW1PD4 135895362 IC50 = 430 nM T96623 CBA73O 135895363 IC50 = 28 nM T96623 CZC4H8 135895364 IC50 = 24 nM T96623 CY0TZ8 135895365 IC50 = 24 nM T96623 C3TYF8 135895374 IC50 = 620 nM T96623 CJ81CD 135895375 IC50 = 160 nM T96623 C3UQ2E 135895376 IC50 > 100000 nM T96623 CNF5H2 135895378 IC50 = 1600 nM T96623 C4FT1I 135895387 IC50 = 250 nM T96623 C36SZT 135911693 IC50 = 37 nM T96623 CJ6N8V 135911694 IC50 = 130 nM T96623 C8DF2L 135911696 IC50 = 184 nM T96623 CQUX92 135911697 IC50 = 163 nM T96623 CA09KE 135911698 IC50 = 85 nM T96623 C29BPD 135911699 IC50 = 190 nM T96623 CXO23J 135911700 IC50 = 214 nM T96623 C60NAD 135911701 IC50 = 26 nM T96623 C8ZV5G 135928046 IC50 = 84 nM T96623 CYQJ21 136002277 IC50 < 5 nM T96623 CFM9A7 136002278 IC50 = 7.4 nM T96623 C7B3FG 136002280 IC50 = 8.8 nM T96623 CLZF76 136002282 IC50 = 230 nM T96623 C7J4LO 136002295 IC50 = 5.4 nM T96623 C0JM6U 136002296 IC50 < 5 nM T96623 CXD7L4 136002297 IC50 < 5 nM T96623 C5SX1H 136002299 IC50 < 5 nM T96623 CQL31N 136002300 IC50 < 5 nM T96623 CRQD18 136002303 IC50 = 24 nM T96623 CF6GV3 136002305 IC50 = 8.6 nM T96623 CY5SE3 136002306 IC50 < 5 nM T96623 CU10GT 136002307 IC50 = 39 nM T96623 C8C2JW 136002308 IC50 = 14 nM T96623 CYO8L7 136002309 IC50 = 34 nM T96623 C4HG7V 136002310 IC50 = 34 nM T96623 CHK34F 136002312 IC50 = 24 nM T96623 C5IW1J 136002313 IC50 = 32 nM T96623 C8KBD3 136002314 IC50 = 32 nM T96623 CV67TM 136002315 IC50 = 22 nM T96623 CWG5C6 136002318 IC50 = 20 nM T96623 C3TY6D 136002319 IC50 = 19 nM T96623 CS4HB2 136002320 IC50 = 22 nM T96623 CT1N0M 136002321 IC50 = 250 nM T96623 C9UE5M 136002322 IC50 = 27 nM T96623 C8WA3J 136002323 IC50 = 40 nM T96623 C4P1FH 136002328 IC50 = 10 nM T96623 C7EZ9A 136002329 IC50 = 36 nM T96623 C6UJ5B 136002330 IC50 = 260 nM T96623 COY05V 136002331 IC50 = 48 nM T96623 CV4HF8 136002332 IC50 = 62 nM T96623 CEQ32X 136002333 IC50 = 33 nM T96623 C7SX3C 136002345 IC50 = 34 nM T96623 CAWT98 136002346 IC50 = 20 nM T96623 CYBR94 136002347 IC50 = 15 nM T96623 CA8X2C 136002348 IC50 < 5 nM T96623 C7PZI2 136002349 IC50 < 5 nM T96623 CU65ZA 136002357 IC50 < 5 nM T96623 C4K6AI 136002365 IC50 < 5 nM T96623 CJ8CU4 136042262 IC50 = 12.6 nM T96623 CQZ42G 136042263 IC50 = 12 nM T96623 C1U5HK 136042264 IC50 = 40 nM T96623 C1N4CU 136082876 Ki = 126 nM T96623 C3ZBM8 136110909 IC50 = 73 nM T96623 CG06VA 136110910 IC50 = 389 nM T96623 C63FBA 136110911 IC50 = 393 nM T96623 CX27KJ 136110912 IC50 = 120 nM T96623 C5GD7K 136110913 IC50 = 143 nM T96623 CHQ05G 136110914 IC50 = 151 nM T96623 C3Y8LO 136110915 IC50 = 1770 nM T96623 CU8T5Q 136110916 IC50 = 446 nM T96623 CG2PO0 136110917 IC50 = 111 nM T96623 CUQ0B5 136110919 IC50 = 126 nM T96623 C1Y5HJ 136110920 IC50 = 68 nM T96623 CFPA47 136110921 IC50 = 384 nM T96623 CU6F1X 136110922 IC50 = 116 nM T96623 CCP4S9 136126672 IC50 = 20000 nM T96623 C2SRX9 136198647 IC50 > 100000 nM T96623 CEX34H 136198648 IC50 > 100000 nM T96623 CN0XY9 136198649 IC50 > 100000 nM T96623 CP79HX 136198650 IC50 > 100000 nM T96623 CR3LD9 136198651 IC50 > 100000 nM T96623 CEWC75 136198653 IC50 > 100000 nM T96623 C1G3FR 136254259 IC50 = 85000 nM T96623 CTCO28 136934953 IC50 > 100000 nM T96623 CMZ90X 136934954 IC50 > 100000 nM T96623 CW40ER 136934955 IC50 > 100000 nM T96623 CKS79P 136934956 IC50 > 100000 nM T96623 CA4OC9 136934957 IC50 > 500000 nM T96623 CI8FR0 136934958 IC50 > 250000 nM T96623 C5VIG4 136934959 IC50 > 100000 nM T96623 C2YZ6E 136934960 IC50 > 100000 nM T96623 C6B4DY 136934961 IC50 > 100000 nM T96623 C01EUC 137069409 IC50 = 108 nM T96623 C0KZD3 137069410 IC50 = 76 nM T96623 COZ20T 137069411 IC50 = 237 nM T96623 C81TKF 137069412 IC50 = 101 nM T96623 C9PDL7 137069413 IC50 = 167 nM T96623 CKH8P9 137069414 IC50 = 1100 nM T96623 CB3P2W 137069415 IC50 = 146 nM T96623 CE35LW 137069416 IC50 = 149 nM T96623 CEL0H2 137069417 IC50 = 160 nM T96623 C7PGC2 137069418 IC50 = 87 nM T96623 CGWX25 137069419 IC50 = 114 nM T96623 CZX7K1 137069420 IC50 = 87 nM T96623 CFOU34 137069421 IC50 = 135 nM T96623 C18RKL 137069422 IC50 = 142 nM T96623 CG05CN 137069423 IC50 = 83 nM T96623 C2GB4N 137069424 IC50 = 35 nM T96623 CYF42G 137069425 IC50 = 99 nM T96623 CTG86A 137069426 IC50 = 141 nM T96623 C4ZM0V 137069427 IC50 = 144 nM T96623 CQEZ48 137069428 IC50 = 736 nM T96623 CZ8IH9 137069429 IC50 = 133 nM T96623 CTI86X 137069430 IC50 = 182 nM T96623 C5GKE7 137069431 IC50 = 636 nM T96623 C1SQD6 137349251 IC50 = 250 nM T96623 C5QI4W 137630301 IC50 = 1500 nM T96623 CH02MW 137630302 IC50 = 3000 nM T96623 CU8QM4 137630303 IC50 = 580 nM T96623 CK0F5U 137630304 IC50 = 460 nM T96623 C4AS7V 137630305 IC50 = 780 nM T96623 C3BA4Y 137630306 IC50 = 370 nM T96623 CHQ2E1 137630307 IC50 = 170 nM T96623 CM9OS6 137630308 IC50 = 1100 nM T96623 CISF34 137630309 IC50 = 1300 nM T96623 CB92LP 137630310 IC50 = 5700 nM T96623 CI0L4Y 137630311 IC50 = 1400 nM T96623 C27KHG 137630312 IC50 = 1300 nM T96623 CM58HC 137630313 IC50 = 610 nM T96623 CALI48 137630314 IC50 = 3400 nM T96623 CJ1HO2 137630315 IC50 = 2500 nM T96623 CPRV51 137630316 IC50 = 580 nM T96623 CX2V9M 137630317 IC50 = 1800 nM T96623 CAG45B 137630318 IC50 = 500 nM T96623 CWIS63 137630319 IC50 = 200 nM T96623 C7SIN2 137630320 IC50 = 350 nM T96623 C0W2IL 137630321 IC50 = 150 nM T96623 C8SL1T 137630322 IC50 = 330 nM T96623 CNMI52 137630323 IC50 = 630 nM T96623 C4LM5I 137630324 IC50 = 390 nM T96623 C6YMZ3 137630325 IC50 = 760 nM T96623 C0L7KO 137630326 IC50 = 2300 nM T96623 CIK9P8 137630327 IC50 = 590 nM T96623 CT2Q6J 137630328 IC50 = 710 nM T96623 CLKY90 137630329 IC50 = 800 nM T96623 C4MQ7W 137630330 IC50 = 680 nM T96623 C7DVE3 137630331 IC50 = 800 nM T96623 CX71WB 137630333 IC50 = 1500 nM T96623 CO8P7F 137630334 IC50 = 980 nM T96623 C8TID9 137630336 IC50 = 2600 nM T96623 CK74TI 137630337 IC50 = 2400 nM T96623 C8O4AS 137630338 IC50 = 1300 nM T96623 C8K0VC 137630339 IC50 = 400 nM T96623 C6ZV3I 137630341 IC50 = 470 nM T96623 CO3E7I 137630342 IC50 = 1900 nM T96623 C2FM8P 137630343 IC50 = 3600 nM T96623 CGB39V 137630344 IC50 = 980 nM T96623 C5L7RV 137630346 IC50 = 740 nM T96623 C4HFT9 137630347 IC50 = 1700 nM T96623 C2K9YN 137630348 IC50 = 570 nM T96623 C4JP3E 137630349 IC50 = 1300 nM T96623 CX2J6Y 137630350 IC50 = 730 nM T96623 CI42JO 137630351 IC50 = 410 nM T96623 CNHA69 137630352 IC50 = 4000 nM T96623 CS86LM 137630353 IC50 = 660 nM T96623 CY41CO 137630355 IC50 = 230 nM T96623 CM91KX 137630356 IC50 = 900 nM T96623 CG8A6F 137630357 IC50 = 1100 nM T96623 CXC82I 137630361 IC50 = 1100 nM T96623 D05GKC 108003 IC50 = 90 nM T96623 D05NWF 6022 IC50 = 42159 nM T96623 D08CZD 3777900 IC50 > 4000000 nM T96623 D0K0TJ 24772860 Ki = 1.1 nM T96623 D0T3PW 5281672 IC50 = 13500 nM T96623 D0T4MS 4369536 IC50 = 25 nM T96623 D0ZA6G 6323491 IC50 = 19 nM T78429 D02RJY 11442891 IC50 > 10000 nM T78429 D02UFQ 11620908 IC50 > 10000 nM T78429 D02ZQS 16095342 IC50 > 10000 nM T78429 D03HUX 49792852 IC50 > 10000 nM T78429 D0E3TC 44259 IC50 = 1 nM T78429 D0O0LS 25141092 IC50 > 10000 nM T78429 D0O6ZO 9952773 IC50 > 10000 nM T78429 D0P1CV 46191454 IC50 > 10000 nM T78429 D0Q9UX 16718576 IC50 > 10000 nM T78429 D0Z5DM 5081913 IC50 = 218 nM T78429 D03BNU 59604787 IC50 > 10000 nM T78429 D01OLO 9820526 Ki = 20 nM T78429 D06WBE 157049 IC50 = 400 nM T78429 D0T3ME 156422 IC50 > 20000 nM T78429 CY58BM 1880 IC50 = 9820 nM T78429 COYW98 9222 IC50 > 667000 nM T78429 C23GZX 327527 IC50 = 2440 nM T78429 CAS18T 359052 IC50 = 7400 nM T78429 C1ZG2U 449087 IC50 > 10000 nM T78429 CYN49L 575802 IC50 = 37900 nM T78429 CU73ST 599501 IC50 > 100000 nM T78429 CR98MZ 613528 IC50 = 2200 nM T78429 CR38XJ 613585 IC50 > 50000 nM T78429 CO13HQ 619692 IC50 = 30000 nM T78429 CPC4Z5 624619 IC50 = 9690 nM T78429 CEAR46 658319 IC50 = 2511.89 nM T78429 CW94YE 700562 IC50 > 30000 nM T78429 C2U5OA 745571 IC50 = 7800 nM T78429 C84ZOX 765847 IC50 = 12700 nM T78429 CRJ8X2 1232489 IC50 = 98600 nM T78429 CX7YE3 1257937 IC50 = 35400 nM T78429 C1SVD2 2132479 IC50 = 4000 nM T78429 C0ZI1F 2756534 IC50 = 1100 nM T78429 CT6P3F 2782903 IC50 = 2600 nM T78429 CMC16L 2782960 IC50 = 22400 nM T78429 C0EC9B 2807839 IC50 = 1584.89 nM T78429 CJWX69 3848929 IC50 > 200000 nM T78429 CE4M1Y 4278270 IC50 = 2900 nM T78429 C2DQY6 5324413 Ki > 30000 nM T78429 CDN4O5 5469267 IC50 = 7300 nM T78429 C8WD6A 6123787 IC50 = 19600 nM T78429 CGYE97 6419765 IC50 = 12.88 nM T78429 C92CUV 6875792 IC50 = 3710 nM T78429 C04EDX 9549298 IC50 = 40 nM T78429 CGH0R4 9796523 IC50 = 23 nM T78429 CD71UI 9813758 IC50 = 150 nM T78429 C6TZ7U 9813880 IC50 = 950 nM T78429 CL4ZD3 9813985 IC50 = 63 nM T78429 C6NGV0 9826896 IC50 = 7000 nM T78429 CI7MW0 9852185 IC50 = 3070 nM T78429 CRC65X 9863786 IC50 > 30000 nM T78429 CM5Z8X 9869943 IC50 = 50000 nM T78429 CHF3I9 9879057 IC50 = 7.943 nM T78429 C18HKQ 9885748 IC50 = 72000 nM T78429 C6MZB1 9900652 IC50 = 58 nM T78429 C3QW5M 9922100 IC50 = 18.2 nM T78429 C3DKI1 9932374 IC50 = 70 nM T78429 CS5KX9 9938299 IC50 > 10000 nM T78429 CK8V5N 9943895 IC50 = 50 nM T78429 CW30AG 9954114 IC50 = 40 nM T78429 C0V7UW 9958506 IC50 > 11000 nM T78429 COET08 9965424 IC50 = 100 nM T78429 C3EP2O 9965828 IC50 = 300 nM T78429 C4IT9O 9985550 IC50 = 45 nM T78429 C6PW4K 9989716 Ki > 30000 nM T78429 CY97GJ 9992352 IC50 = 2200 nM T78429 C2D4IZ 10007960 IC50 = 51 nM T78429 CWK19D 10008543 IC50 = 107 nM T78429 CXS2Z8 10018040 IC50 = 750 nM T78429 C63LXA 10038414 IC50 = 4100 nM T78429 C7YD1X 10048045 IC50 > 10000 nM T78429 C2GTX0 10076485 IC50 = 27 nM T78429 C1ZR5V 10098997 IC50 = 70 nM T78429 CW59RK 10109125 IC50 = 45.71 nM T78429 CMP0W2 10117126 IC50 = 34 nM T78429 C9ARB8 10126159 IC50 = 170 nM T78429 CU4F6P 10215156 IC50 = 19 nM T78429 CT58NL 10220851 IC50 = 25.12 nM T78429 CK0SI6 10242687 IC50 = 4700 nM T78429 CSGD16 10246246 IC50 = 41 nM T78429 C9JS8K 10257503 IC50 = 48 nM T78429 C6MY7H 10298332 IC50 = 47 nM T78429 CT13WV 10334531 IC50 = 2500 nM T78429 CDU19Z 10346473 IC50 = 477 nM T78429 CNTK08 10355567 IC50 = 5800 nM T78429 C30VJZ 10361228 IC50 = 1300 nM T78429 CFP54N 10399267 IC50 = 2000 nM T78429 CF9MV3 10410982 IC50 = 66 nM T78429 CKU7Z3 10424325 IC50 = 2400 nM T78429 C7HBP6 10429593 IC50 > 10000 nM T78429 CE3L7Z 10459074 IC50 = 589 nM T78429 CYKG01 10461267 IC50 = 1.9 nM T78429 C95PCE 10473450 IC50 = 1400 nM T78429 C4MAH5 10564173 IC50 = 1100 nM T78429 C8G3UE 10805474 IC50 = 14000 nM T78429 C4ZV5I 11149107 IC50 = 5011.87 nM T78429 CRP61Y 11156148 IC50 = 398.11 nM T78429 CJ7U4I 11161778 IC50 = 10.96 nM T78429 CNCT02 11173949 IC50 = 6 nM T78429 CW5C9X 11186250 IC50 = 158.49 nM T78429 C9GY2P 11207091 IC50 = 1584.89 nM T78429 CT19ID 11207978 IC50 = 316.23 nM T78429 C6C3JX 11281930 IC50 > 10000 nM T78429 CBOP58 11293798 Ki = 340 nM T78429 C9TOG5 11304835 IC50 = 19.95 nM T78429 C9CWY7 11323357 IC50 = 501.19 nM T78429 C5HC6S 11336070 IC50 = 130 nM T78429 CV43QF 11336440 IC50 = 501.19 nM T78429 CM0GX5 11350427 IC50 = 25.12 nM T78429 C26BZX 11362471 Ki = 380 nM T78429 CWXB93 11397177 Ki > 10000 nM T78429 CU76FI 11402873 IC50 = 2511.89 nM T78429 C0APW4 11422034 IC50 > 10000 nM T78429 CVX70O 11427162 IC50 = 501.19 nM T78429 C8VT9G 11436911 IC50 = 1584.89 nM T78429 CMVN46 11438476 IC50 = 333 nM T78429 C7X4HG 11448486 IC50 = 28 nM T78429 CM21YJ 11453049 IC50 = 12.59 nM T78429 CJC95A 11454205 IC50 > 10000 nM T78429 CPL1G0 11492368 IC50 = 36200 nM T78429 C2FVI1 11496203 IC50 = 500 nM T78429 CY1A6E 11499932 IC50 > 23500 nM T78429 C8LE9Y 11507173 IC50 = 6300 nM T78429 CTZP60 11507891 IC50 = 8200 nM T78429 CP94UI 11521540 IC50 = 6600 nM T78429 C7HMO6 11526786 IC50 > 10000 nM T78429 CTG83F 11539329 Ki > 3200 nM T78429 CY8D0L 11550419 IC50 = 18000 nM T78429 CD84CQ 11550651 IC50 = 4600 nM T78429 C5TI2K 11555269 IC50 = 7.943 nM T78429 CBK97Y 11558904 IC50 = 20160 nM T78429 C4XKL7 11559659 IC50 = 4060 nM T78429 CM9TL3 11564688 IC50 = 35700 nM T78429 C28EAJ 11568801 IC50 = 50 nM T78429 C7QDV6 11579568 IC50 = 12700 nM T78429 CEZC37 11579690 IC50 = 5000 nM T78429 CO9KP5 11583459 IC50 > 10000 nM T78429 CWTV61 11588556 IC50 = 19000 nM T78429 CMIL86 11590363 Ki > 3200 nM T78429 CULP46 11598695 IC50 = 31.62 nM T78429 CK6Y0A 11608156 IC50 = 19900 nM T78429 CJP83V 11608384 IC50 = 10600 nM T78429 C1KG7N 11608463 IC50 = 25800 nM T78429 CH7P9Z 11608743 IC50 = 8000 nM T78429 C93QIF 11611619 IC50 = 7.943 nM T78429 CRY7Z9 11615418 IC50 = 4700 nM T78429 C93UKS 11617172 IC50 = 19 nM T78429 C1P5BA 11623540 IC50 > 35000 nM T78429 CO2JL0 11625181 IC50 < 15848.93 nM T78429 CGX96V 11626927 IC50 > 15848.93 nM T78429 CIZ5E8 11631150 IC50 = 3400 nM T78429 CKZ84S 11637076 IC50 > 32500 nM T78429 C9T6SC 11640926 Ki > 3200 nM T78429 C2F8XO 11641780 IC50 = 7.943 nM T78429 CKC09N 11643997 IC50 > 667000 nM T78429 C4PA7Q 11651984 IC50 = 10300 nM T78429 C9TLI8 11651993 IC50 = 50 nM T78429 C3PVG1 11653077 IC50 = 13000 nM T78429 C1V5TK 11658697 IC50 = 13900 nM T78429 CVRY32 11658724 IC50 > 50000 nM T78429 C7NWM0 11667571 IC50 = 40 nM T78429 CDMF06 11672971 IC50 = 6300 nM T78429 CY92SG 11680280 IC50 = 14000 nM T78429 CJ9KN7 11683817 IC50 > 10000 nM T78429 CDSB23 11688891 IC50 = 58000 nM T78429 CU0E8O 11690457 Ki > 10000 nM T78429 CVFY45 11694530 IC50 > 27500 nM T78429 CK70RY 11694599 IC50 = 2500 nM T78429 CEA5G8 11701554 IC50 > 49000 nM T78429 C6CD2A 11702259 IC50 > 39500 nM T78429 CM48EL 11702815 IC50 = 5600 nM T78429 CB0AP2 11705863 Ki > 10000 nM T78429 CDE89K 11705934 IC50 = 10 nM T78429 CO8XH4 11719652 IC50 = 20 nM T78429 C45EWD 11723489 IC50 = 120 nM T78429 CTKJ45 11757505 IC50 = 54 nM T78429 C05ANW 11778364 IC50 = 15100 nM T78429 C9JT4S 11847343 IC50 > 10000 nM T78429 CZTR57 11954411 IC50 = 1670 nM T78429 C8E4TS 11992146 IC50 > 200000 nM T78429 CG7X9F 12330558 IC50 > 100000 nM T78429 C8TCR5 13297340 IC50 = 7400 nM T78429 C3QKT4 14355186 Ki > 30000 nM T78429 CRKG41 15944053 IC50 > 200000 nM T78429 CYW2V4 15944061 IC50 > 200000 nM T78429 C2DKR4 15979284 IC50 = 100 nM T78429 CVB2D9 16004583 IC50 = 64300 nM T78429 CS8P1W 16004585 IC50 = 54700 nM T78429 CFPW41 16007116 Ki > 3100 nM T78429 C9TU1O 16046126 IC50 > 1000 nM T78429 CPJ94T 16047031 IC50 = 158.49 nM T78429 C1Y0VG 16047033 IC50 = 398.11 nM T78429 CD1OQ4 16047143 IC50 = 650 nM T78429 C1MA4Q 16047147 IC50 = 1584.89 nM T78429 CXV5E7 16047740 IC50 = 158.49 nM T78429 CAPR-79 16047856 IC50 = 199.53 nM T78429 CJI9Z4 16047968 IC50 = 251.19 nM T78429 C2J6PS 16048084 IC50 = 630.96 nM T78429 C6N5YF 16048085 IC50 = 251.19 nM T78429 CM21OB 16048194 IC50 = 1584.89 nM T78429 CYQO76 16048303 IC50 = 1584.89 nM T78429 CTI58R 16048308 IC50 = 1584.89 nM T78429 C1QJ3P 16048414 IC50 = 3981.07 nM T78429 C6EU9X 16048415 IC50 = 3981.07 nM T78429 C2W0CV 16048543 IC50 = 7943.28 nM T78429 CL1NQ5 16048544 IC50 = 7943.28 nM T78429 CKV4G1 16079040 IC50 = 1100 nM T78429 C7Z4LV 16095343 IC50 > 10000 nM T78429 C10VKP 16105041 IC50 = 24160 nM T78429 CB8H0X 16663529 IC50 = 18 nM T78429 CUR7H3 16719862 IC50 > 200000 nM T78429 CF0H3L 17229016 IC50 = 60100 nM T78429 C9JVQ0 17930948 IC50 = 39.81 nM T78429 CT7OC2 20767724 IC50 = 10.96 nM T78429 CE7AV5 20767725 IC50 = 34.67 nM T78429 C0T2VF 20823920 IC50 = 490 nM T78429 CX0E5L 20823952 IC50 = 290 nM T78429 CKQV75 20823956 IC50 = 190 nM T78429 C9CUN2 20823959 IC50 = 370 nM T78429 CD1K8E 20823960 IC50 = 27 nM T78429 C1FE5V 20823975 IC50 = 40 nM T78429 CG4H7B 20823982 IC50 = 95 nM T78429 C9W2GS 20823986 IC50 = 290 nM T78429 CKTI83 20823993 IC50 = 85 nM T78429 C6A3PV 20823995 IC50 = 360 nM T78429 CO27KL 20823998 IC50 > 1000 nM T78429 C2S7RG 20824041 IC50 = 520 nM T78429 C9O4WF 20824060 IC50 = 260 nM T78429 CXG6R2 21083789 IC50 = 180 nM T78429 CS1MB4 21083790 IC50 = 26 nM T78429 C7NMQ8 21083887 IC50 = 9 nM T78429 CP14LT 21083893 IC50 = 53 nM T78429 CYC65I 21083894 IC50 = 32 nM T78429 CA61QF 21083895 IC50 = 22 nM T78429 C8WUE9 21083896 IC50 = 5 nM T78429 CE20HN 21083898 IC50 = 210 nM T78429 CWIR51 21083902 IC50 = 81 nM T78429 CWTV36 21083906 IC50 = 38.9 nM T78429 C9YMR6 21083908 IC50 = 2500 nM T78429 C40AEJ 22285027 IC50 = 23 nM T78429 C14NDQ 22291467 IC50 = 1340 nM T78429 CB9F8U 22291471 IC50 = 348 nM T78429 CZYW61 22291566 IC50 = 146 nM T78429 CBJL25 22291634 IC50 = 297 nM T78429 CEXB18 22291652 IC50 = 1.6 nM T78429 C1UKQ5 22291682 IC50 = 29 nM T78429 CX31HI 22291687 IC50 = 19 nM T78429 CW6RL1 22291691 IC50 = 10 nM T78429 CW59EG 22291701 IC50 = 1250 nM T78429 CUD21A 22291734 IC50 = 90 nM T78429 C3AXH0 22291741 IC50 = 612 nM T78429 CGV16P 22291750 IC50 = 40 nM T78429 C73AZU 22291899 IC50 = 210 nM T78429 C7Y0VE 22291924 IC50 = 125 nM T78429 CZE23T 22291961 IC50 = 33 nM T78429 C5JH1P 22477600 IC50 = 3162.28 nM T78429 C7C1YA 23400922 IC50 = 72 nM T78429 C5UW7F 23400928 IC50 = 630 nM T78429 C6JV7W 23400934 IC50 = 570 nM T78429 CK54QC 23400993 IC50 = 1300 nM T78429 C8OFA1 23400995 IC50 = 150 nM T78429 CD5S7O 23401001 IC50 = 280 nM T78429 CVX51K 23401012 IC50 = 98 nM T78429 CTR87W 23401015 IC50 = 120 nM T78429 C8Y5VA 23401016 IC50 = 520 nM T78429 C32GJX 23586307 IC50 = 240 nM T78429 CC21PY 23648887 IC50 = 199.53 nM T78429 CMD65I 23648890 IC50 = 39.81 nM T78429 C4C2XA 23648920 IC50 = 251.19 nM T78429 CWX53C 23648921 IC50 = 316.23 nM T78429 C2R1QH 23648953 IC50 = 79.43 nM T78429 CBA39U 23657350 IC50 = 12.88 nM T78429 CDMI50 23661564 IC50 > 200000 nM T78429 CJM4C7 24219848 IC50 > 100000 nM T78429 C7YG1N 24759534 IC50 = 55000 nM T78429 C2UOE0 24766030 IC50 > 50000 nM T78429 CLBP72 24798571 IC50 = 24689 nM T78429 C9PA0M 24807809 IC50 > 10000 nM T78429 CCP2M3 24822704 IC50 > 50000 nM T78429 CQN3Z7 24825710 IC50 = 9 nM T78429 C8OUR0 24856835 IC50 = 630.96 nM T78429 C13QYB 24884503 IC50 > 2000 nM T78429 CJ7XN5 24896721 IC50 > 50000 nM T78429 CDHC95 24896725 IC50 > 50000 nM T78429 CY8L7E 24896769 IC50 > 10000 nM T78429 CP3M7W 24898267 IC50 > 50000 nM T78429 CG51ON 24898486 IC50 > 50000 nM T78429 C78VZS 24898709 IC50 > 50000 nM T78429 CM0FP2 24944518 IC50 = 10 nM T78429 CLZ23U 24951610 IC50 > 30000 nM T78429 C7N4DI 24959043 IC50 = 1100 nM T78429 C6CVK4 24959046 IC50 = 200 nM T78429 C97XGO 24959409 IC50 = 330 nM T78429 CX03EC 24959770 IC50 = 20000 nM T78429 C8UK3G 24959772 IC50 = 2000 nM T78429 CO60FQ 24960141 IC50 = 1900 nM T78429 CH3D1L 24960509 IC50 = 2400 nM T78429 CUA17W 24961607 IC50 = 1400 nM T78429 CWE0L7 24983829 IC50 = 19.95 nM T78429 C2O0QA 24984297 IC50 = 10 nM T78429 CH32GJ 24984615 IC50 = 316.23 nM T78429 C5RY8D 24984616 IC50 = 63.1 nM T78429 C90YFT 24984774 IC50 = 19.95 nM T78429 CM3EI4 24984940 IC50 = 19.95 nM T78429 CQ2Z7T 24985115 IC50 = 199.53 nM T78429 C8O0JE 24985283 IC50 = 19.95 nM T78429 C4EG8R 24993189 IC50 > 10000 nM T78429 C67FGO 25071914 IC50 = 12.59 nM T78429 C90QPI 25093427 IC50 = 230 nM T78429 CHTR48 25093428 IC50 = 28.84 nM T78429 CTD7L0 25093430 IC50 = 2.512 nM T78429 CSX0O1 25093431 IC50 = 10 nM T78429 C9AIZ8 25093432 IC50 = 190 nM T78429 C2S5GF 25093433 IC50 = 140 nM T78429 CQEP18 25093434 IC50 = 270 nM T78429 CMJ8E0 25093435 IC50 = 280 nM T78429 CW92XG 25093436 IC50 = 44 nM T78429 C8CJQ9 25093437 IC50 = 95 nM T78429 CXM5Q4 25093438 IC50 = 130 nM T78429 C9Y3PO 25093439 IC50 = 7.943 nM T78429 CNE20C 25093440 IC50 = 22.91 nM T78429 C48WIP 25093441 IC50 = 21 nM T78429 CJL3O1 25093442 IC50 = 230 nM T78429 CH27WL 25093443 IC50 = 8 nM T78429 C6FEC5 25093444 IC50 = 38.02 nM T78429 CN52FS 25093445 IC50 = 42.66 nM T78429 CU5CK2 25093446 IC50 = 3 nM T78429 C2YXB7 25093447 IC50 = 23 nM T78429 C6KFE7 25093448 IC50 = 44.67 nM T78429 COC9K8 25093449 IC50 = 21 nM T78429 C0N9GE 25093450 IC50 = 18.2 nM T78429 CR81QD 25093451 IC50 = 7 nM T78429 CRX17M 25093452 IC50 = 51 nM T78429 CS1MO6 25093453 IC50 = 8 nM T78429 CT41VL 25093454 IC50 < 9 nM T78429 CYC24O 25093455 IC50 = 19 nM T78429 CU45OM 25093456 IC50 = 12.88 nM T78429 C52VZG 25093457 IC50 = 26.92 nM T78429 CO58WP 25093458 IC50 = 14 nM T78429 C6P0DN 25093459 IC50 = 36.31 nM T78429 CD7WE8 25093460 IC50 = 590 nM T78429 C2KY1G 25094210 IC50 > 10000 nM T78429 C34MQJ 25137988 IC50 = 416.87 nM T78429 CKT3M0 25137989 IC50 = 195 nM T78429 C7UXT9 25137990 IC50 = 465 nM T78429 CIA60B 25137991 IC50 = 563 nM T78429 C52FXY 25137992 IC50 = 331 nM T78429 C1D0MV 25137993 IC50 = 620 nM T78429 CR08TY 25137994 IC50 = 1010 nM T78429 CIWD80 25137995 IC50 = 716 nM T78429 CWV3C2 25137996 IC50 = 303 nM T78429 CNWC59 25137997 IC50 = 263.03 nM T78429 CXNY85 25137998 IC50 = 709 nM T78429 CTWA47 25137999 IC50 > 20000 nM T78429 C2RU5P 25138000 IC50 = 557 nM T78429 CYJ31L 25138001 IC50 = 1850 nM T78429 C6VE4L 25138002 IC50 = 704 nM T78429 C5CT2M 25138003 IC50 = 964 nM T78429 CW84BS 25138004 IC50 = 980 nM T78429 C8RF2Z 25138005 IC50 = 1880 nM T78429 CG98XL 25138006 IC50 = 4400 nM T78429 C2LAU0 25138007 IC50 = 454 nM T78429 C6BWZ8 25145145 IC50 > 100 nM T78429 C78YWA 25145716 IC50 > 500 nM T78429 C6Q1ST 25169524 IC50 = 250 nM T78429 CF4H8C 25190912 IC50 < 15848.93 nM T78429 CYG76T 25190913 IC50 < 15848.93 nM T78429 CMQ32Y 25190914 IC50 < 15848.93 nM T78429 C4D3FJ 25190920 IC50 = 15848.93 nM T78429 C1LZ2V 25190921 IC50 > 15848.93 nM T78429 CY9GT4 25190922 IC50 > 15848.93 nM T78429 CQMR47 25190923 IC50 > 15848.93 nM T78429 C5M8HZ 25190924 IC50 > 15848.93 nM T78429 CE8X6M 25190925 IC50 > 15848.93 nM T78429 CF6Z9S 25190926 IC50 > 15848.93 nM T78429 CUZ2N7 25190927 IC50 > 15848.93 nM T78429 C6FGQ1 25206346 IC50 = 8100 nM T78429 CNG96H 25210579 IC50 > 10000 nM T78429 CRO09K 25211064 IC50 = 9170 nM T78429 C56VHY 25219675 IC50 > 100000 nM T78429 CT9IN1 25263282 IC50 = 33.88 nM T78429 CN5E0F 25263283 IC50 = 520 nM T78429 CW18IA 25263284 IC50 = 920 nM T78429 CE1GP2 25263285 IC50 = 1500 nM T78429 CQ9X4U 25263286 IC50 = 300 nM T78429 CXN0J8 25263287 IC50 = 33 nM T78429 C37JSG 25263288 IC50 = 15 nM T78429 CI7PA9 25263289 IC50 = 15 nM T78429 CIUH13 25263290 IC50 = 160 nM T78429 CWP6H9 25263291 IC50 = 15 nM T78429 CPC7D9 25263292 IC50 = 33 nM T78429 CB7M1Z 25263293 IC50 = 75 nM T78429 CNH56T 25263294 IC50 = 56 nM T78429 C1Z6QP 25263295 IC50 = 25 nM T78429 C02XNR 25263296 IC50 = 16 nM T78429 CM0EF4 42618139 IC50 = 1258.93 nM T78429 CWS37O 42618140 IC50 = 100 nM T78429 CQE43D 42618141 IC50 = 398.11 nM T78429 C2IK0N 42618142 IC50 = 794.33 nM T78429 C2JV3O 42618143 IC50 = 125.89 nM T78429 CG01BO 42618144 IC50 = 100 nM T78429 CCSQ57 42618145 IC50 = 398.11 nM T78429 CW7X6L 42618146 IC50 = 5011.87 nM T78429 C4K6PD 42618147 IC50 = 12589.25 nM T78429 C5SL3N 42618148 IC50 = 3162.28 nM T78429 CYU47O 42618149 IC50 = 1258.93 nM T78429 CWD4R1 42618150 IC50 = 1995.26 nM T78429 C5X2UV 42618151 IC50 = 1000 nM T78429 CIN5U6 42618152 IC50 = 5011.87 nM T78429 CW8VP1 42618153 IC50 = 630.96 nM T78429 CCB0L2 42618154 IC50 = 158.49 nM T78429 CC7GS2 42618155 IC50 = 794.33 nM T78429 CZ86OF 42618156 IC50 = 158.49 nM T78429 CX9N3L 42618157 IC50 = 1258.93 nM T78429 C38FZM 42618158 IC50 = 630.96 nM T78429 C2I7HC 42618159 IC50 = 1258.93 nM T78429 C6YSW0 42618160 IC50 = 19952.62 nM T78429 C3IY4O 42618161 IC50 = 3981.07 nM T78429 C1CY8R 42618162 IC50 = 5011.87 nM T78429 C80KDA 42618163 IC50 = 7943.28 nM T78429 CG28AW 42618164 IC50 = 3162.28 nM T78429 CU9E4P 42629114 IC50 > 10000 nM T78429 CO4FV0 42630578 IC50 = 39.81 nM T78429 C90BUF 43157763 IC50 = 75700 nM T78429 CJ7D5T 43157843 IC50 > 100000 nM T78429 C6Z2SA 43560957 IC50 = 88000 nM T78429 CNO13E 44127365 IC50 = 7060 nM T78429 CXBT98 44127366 IC50 = 4750 nM T78429 CO42DC 44138048 IC50 > 10000 nM T78429 CL65QV 44138049 IC50 > 10000 nM T78429 CLW80F 44160269 IC50 = 1000 nM T78429 C6RN7P 44187181 IC50 = 7.079 nM T78429 CI4Y7O 44187182 IC50 = 7.079 nM T78429 C6LTC3 44187183 IC50 = 12.02 nM T78429 CEL61X 44229839 IC50 > 10000 nM T78429 CYE36B 44241613 IC50 > 40000 nM T78429 C6LG5T 44241614 IC50 > 40000 nM T78429 CMI34Q 44353870 IC50 = 26 nM T78429 CSEY31 44353885 IC50 = 155 nM T78429 CR13ES 44353890 IC50 = 512.86 nM T78429 CI3U0J 44353891 IC50 = 309 nM T78429 CA16WX 44353923 IC50 = 146 nM T78429 CIJ19R 44353953 IC50 = 47.86 nM T78429 CCLG72 44353954 IC50 = 59 nM T78429 CO97FH 44353955 IC50 = 60 nM T78429 C86QXB 44353966 IC50 = 214 nM T78429 C15JMN 44353967 IC50 = 269 nM T78429 CLV7G6 44353968 IC50 = 331 nM T78429 C8RZV9 44353969 IC50 = 148 nM T78429 CN91IA 44353987 IC50 = 145 nM T78429 CGB6I4 44353995 IC50 = 10.96 nM T78429 CJIC08 44353996 IC50 = 31 nM T78429 C7MS0Y 44353999 IC50 = 83 nM T78429 CW5J2M 44354000 IC50 = 91 nM T78429 CY6K7E 44354001 IC50 = 91 nM T78429 CFO54D 44354009 IC50 = 117 nM T78429 C7HBR2 44354029 IC50 = 42.66 nM T78429 CJD42L 44354030 IC50 = 43.65 nM T78429 CGDH37 44382918 IC50 > 20000 nM T78429 CS65GI 44382922 IC50 > 20000 nM T78429 CL47KA 44382930 IC50 > 20000 nM T78429 CW8F5K 44383326 IC50 > 20000 nM T78429 CPQE37 44392957 IC50 > 20 nM T78429 CS7N9Y 44406379 IC50 = 200 nM T78429 CEA0O3 44406380 IC50 > 100000 nM T78429 CAW8D0 44406386 IC50 = 400 nM T78429 C9LVS2 44406419 IC50 = 40 nM T78429 CW5YP1 44406467 IC50 = 2200 nM T78429 CRC9U2 44406468 IC50 = 900 nM T78429 COQ56E 44406470 IC50 = 600 nM T78429 C4HSU0 44406486 IC50 = 600 nM T78429 C29MVP 44406487 IC50 = 1000 nM T78429 C47WRS 44406506 IC50 > 100000 nM T78429 CS60YA 44406549 IC50 = 150 nM T78429 C1GJF8 44406564 IC50 = 90 nM T78429 CG5T2C 44406565 IC50 = 39.81 nM T78429 CM58DH 44406581 IC50 = 150 nM T78429 CG3CW4 44406586 IC50 = 60 nM T78429 CPR69I 44406614 IC50 = 50 nM T78429 C1IT5S 44406634 IC50 = 50 nM T78429 C51NLK 44406635 IC50 = 25 nM T78429 CMX18H 44406636 IC50 = 100 nM T78429 CL7M1J 44425584 IC50 = 1000 nM T78429 C2C5OI 44425585 IC50 = 316.23 nM T78429 CZ67YJ 44425588 IC50 = 316.23 nM T78429 C9KTQ7 44425594 IC50 = 158.49 nM T78429 CXV8D5 44425596 IC50 = 251.19 nM T78429 CI26BP 44425599 IC50 = 316.23 nM T78429 C1GY8L 44425606 IC50 = 251.19 nM T78429 COPG94 44427519 IC50 = 5800 nM T78429 CMN54H 44442024 IC50 = 450 nM T78429 C6T7RE 44448365 IC50 = 540 nM T78429 C6LN2Y 44448366 IC50 = 600 nM T78429 CWM3V0 44448369 IC50 = 410 nM T78429 CX4M1T 44448398 IC50 = 380 nM T78429 CCWD87 44448400 IC50 = 8912.51 nM T78429 CL15GU 44448434 IC50 = 8900 nM T78429 CVSP28 44448438 IC50 = 1500 nM T78429 C0HML9 44448550 IC50 = 990 nM T78429 C0VS4B 44448553 IC50 = 230 nM T78429 CL2U8A 44448587 IC50 = 398.11 nM T78429 C1I5OF 44448662 IC50 = 270 nM T78429 C01RDH 44448700 IC50 = 128.82 nM T78429 CA97WK 44448903 IC50 = 3600 nM T78429 C4HQW0 44448967 IC50 = 2500 nM T78429 C2H7WO 44449023 IC50 = 700 nM T78429 CQ1BO7 44449045 IC50 = 440 nM T78429 C9IGA2 44449047 IC50 = 407.38 nM T78429 CJ06YF 44449187 IC50 = 6025.6 nM T78429 CN0K9Q 44449188 IC50 = 64 nM T78429 CH6ND3 44449215 IC50 = 4000 nM T78429 CA78EV 44573281 IC50 = 280 nM T78429 CB4T0A 44583737 IC50 = 3520 nM T78429 C3B9XA 44591531 IC50 = 32.36 nM T78429 CVI6S3 44591532 IC50 = 39.81 nM T78429 C06RIF 44591552 IC50 = 158.49 nM T78429 CCD3F9 44591553 IC50 = 5011.87 nM T78429 CXP21B 44591574 IC50 = 15.85 nM T78429 C4T8XR 44591575 IC50 = 19.95 nM T78429 CHQR35 44591576 IC50 = 39.81 nM T78429 C5Z3LI 44591740 IC50 = 13000 nM T78429 C9JC8E 44608984 IC50 = 4200 nM T78429 C0LSF6 44609136 IC50 = 4800 nM T78429 C0LS2M 44609137 IC50 = 2300 nM T78429 CDK6W9 44609616 IC50 = 3000 nM T78429 CKA93D 44609618 IC50 = 4600 nM T78429 CW5Z2E 44610076 IC50 = 2700 nM T78429 CUQ1B3 44610231 IC50 = 11000 nM T78429 CU3RF1 45139989 IC50 > 10000 nM T78429 CQGZ06 45139991 IC50 > 10000 nM T78429 CW4LQ3 45267192 IC50 = 25.12 nM T78429 C29EIZ 45268050 IC50 = 38.9 nM T78429 CAXI74 45268940 IC50 = 21.88 nM T78429 CST87Y 45269780 IC50 = 14 nM T78429 C87FEM 45270051 IC50 > 40000 nM T78429 C2JVA4 45270368 IC50 = 79 nM T78429 CCNU16 45270611 IC50 = 10.96 nM T78429 CL45SW 45271427 IC50 = 42.66 nM T78429 C1SAJ4 45272329 IC50 = 7.943 nM T78429 CX0A2G 45273193 IC50 = 43.65 nM T78429 CU53FK 45273505 IC50 > 40000 nM T78429 C6E2SC 45482700 IC50 > 10000 nM T78429 CZXH74 45482750 IC50 > 10000 nM T78429 CD2RL3 45485717 IC50 = 6600 nM T78429 CV6N1O 45485718 IC50 = 5100 nM T78429 CS6E2W 45485728 IC50 = 2900 nM T78429 C4BK0A 45485729 IC50 > 50000 nM T78429 CK9FX6 45485737 IC50 = 2400 nM T78429 CC0TY4 45485747 IC50 = 2000 nM T78429 CDPG79 45485755 IC50 = 680 nM T78429 C3T2IE 45485760 IC50 = 1300 nM T78429 CY7QG4 45485771 IC50 = 2500 nM T78429 COH31M 45485772 IC50 = 680 nM T78429 C4A7DL 45485790 IC50 = 10800 nM T78429 CN2Q1J 45485791 IC50 = 7800 nM T78429 CAJ4T7 45485795 IC50 = 16900 nM T78429 CM6C4Y 45485796 IC50 = 680 nM T78429 CNP23F 45485813 IC50 = 2000 nM T78429 CXH2I4 45485814 IC50 = 6000 nM T78429 C4D3MG 45485818 IC50 = 8500 nM T78429 CKR01C 45486822 IC50 = 140 nM T78429 C4OS7C 45486857 IC50 = 1450 nM T78429 CTA0B6 45486858 IC50 = 1950 nM T78429 CUM43N 45486885 IC50 = 590 nM T78429 C5XN7B 45486896 IC50 = 500 nM T78429 CUA97D 46209401 IC50 = 3700 nM T78429 CG7UB8 46229347 IC50 = 5910 nM T78429 CJ89TK 46229373 IC50 = 17300 nM T78429 CY9JA3 46229374 IC50 = 2320 nM T78429 C1DQ5O 46229375 IC50 = 3210 nM T78429 CS05GT 46229376 IC50 = 14200 nM T78429 CNS6V2 46229404 IC50 = 16200 nM T78429 CK7U0P 46229456 IC50 = 52 nM T78429 C75BTR 46229457 IC50 = 98 nM T78429 CI8WA4 46229458 IC50 = 46 nM T78429 C7ON5A 46233287 IC50 > 10000 nM T78429 COTJ39 46863083 IC50 > 30000 nM T78429 C7H4YM 46865419 IC50 > 10000 nM T78429 C5Y4IF 46871625 IC50 = 510 nM T78429 CH43YM 46871627 IC50 = 510 nM T78429 C6PZM5 46871628 IC50 = 420 nM T78429 CJOM49 46880136 IC50 > 50000 nM T78429 C3MKH0 46890182 IC50 = 1430 nM T78429 CR4YS0 46890183 IC50 = 10 nM T78429 C9MFG6 46890212 IC50 = 1360 nM T78429 CRQ86Z 46890213 IC50 = 1790 nM T78429 CO98EK 46890255 IC50 = 310 nM T78429 C09SJD 46890256 IC50 = 1600 nM T78429 CPLG75 46890257 IC50 = 1940 nM T78429 CHN84Z 46890284 IC50 = 8250 nM T78429 C68VPZ 46890285 IC50 = 1570 nM T78429 CI7XG4 46890286 IC50 = 1110 nM T78429 CX5GC1 46890287 IC50 = 280 nM T78429 CA5LG2 46890317 IC50 = 2230 nM T78429 CV9G5B 46890318 IC50 = 180 nM T78429 C2GR4F 46890319 IC50 = 790 nM T78429 C4IA2J 46890320 IC50 = 230 nM T78429 CWD7I0 46890387 IC50 = 170 nM T78429 CGOX07 46890388 IC50 = 620 nM T78429 CJ9L4A 46890389 IC50 = 130 nM T78429 CY07KX 46890390 IC50 = 1220 nM T78429 CVNH70 46933383 IC50 = 47 nM T78429 CQR9K1 46933384 IC50 = 55 nM T78429 CHSF07 49806372 IC50 > 1000 nM T78429 CF91RS 49843531 IC50 > 10000 nM T78429 C83VHI 49864785 IC50 = 590 nM T78429 CV9F6R 49864786 IC50 = 2400 nM T78429 CHU3P4 49864787 IC50 > 30000 nM T78429 C51LGH 49864788 IC50 = 4000 nM T78429 C5KVG1 49864848 IC50 = 11000 nM T78429 CP60MT 49864849 IC50 > 30000 nM T78429 C2UTK6 49864850 IC50 = 320 nM T78429 C3EDR7 49864894 IC50 = 10000 nM T78429 CT9L5E 49864895 IC50 = 14000 nM T78429 COB6T8 49864896 IC50 = 5600 nM T78429 C38LWN 49864897 IC50 = 18000 nM T78429 CZ6C3F 49864932 IC50 > 30000 nM T78429 CO93WA 49864933 IC50 > 30000 nM T78429 CX48UC 49864934 IC50 > 30000 nM T78429 CR1AZ3 49864935 IC50 > 30000 nM T78429 CPAL30 49864982 IC50 = 2100 nM T78429 CL1WH4 49864983 IC50 = 8900 nM T78429 CATJ67 49864984 IC50 > 30000 nM T78429 CYRP85 49865034 IC50 > 30000 nM T78429 C0Y3DJ 49865035 IC50 > 30000 nM T78429 C58HZE 49865036 IC50 > 30000 nM T78429 CX9N0E 49865037 IC50 = 27000 nM T78429 C70NBH 49865092 IC50 > 30000 nM T78429 CZY6D1 49865093 IC50 = 14000 nM T78429 CFOC84 49865094 IC50 = 1300 nM T78429 C0RWA8 49865095 IC50 = 270 nM T78429 CB7YV6 49865096 IC50 = 200 nM T78429 C5ZWS0 49865152 IC50 = 330 nM T78429 CAE53W 49865153 IC50 = 190 nM T78429 C9KOH8 49865154 IC50 = 3700 nM T78429 CRL53S 49865210 IC50 = 550 nM T78429 CY9IX5 49865211 IC50 = 11000 nM T78429 CXQ7W8 49865212 IC50 = 3000 nM T78429 C7JY8O 49865213 IC50 = 380 nM T78429 CVYL14 49865274 IC50 = 530 nM T78429 CU56MF 49865275 IC50 = 7100 nM T78429 CL82UA 49865276 IC50 > 30000 nM T78429 C2KS7B 49865277 IC50 > 30000 nM T78429 CF5B1D 49865328 IC50 = 79 nM T78429 CI2R8J 49865329 IC50 = 310 nM T78429 CG4TE7 49865330 IC50 = 73 nM T78429 C9NS1I 49865383 IC50 = 5100 nM T78429 CL4BG7 49865384 IC50 = 160 nM T78429 CGE56K 49865385 IC50 = 100 nM T78429 CY7Q4W 49865433 IC50 = 140 nM T78429 CUJ47K 49865434 IC50 = 110 nM T78429 C46QLF 49865574 IC50 = 2800 nM T78429 C7D8SP 50905014 IC50 = 16 nM T78429 C2Y6QS 50938552 IC50 > 10000 nM T78429 CH2I3A 50941935 IC50 = 19 nM T78429 CIB60D 50941936 IC50 = 6 nM T78429 C2KE0Y 50941937 IC50 = 13 nM T78429 CAZQ43 51003133 IC50 > 1000 nM T78429 C4NLQ1 51003477 IC50 = 17 nM T78429 C9NYP4 51036677 IC50 > 10000 nM T78429 C4WRY3 51037112 IC50 > 10000 nM T78429 CRI28Z 51037948 IC50 > 10000 nM T78429 CP91XJ 51346795 IC50 = 1700 nM T78429 CXA03W 52920796 IC50 > 100 nM T78429 CE7JI9 52941456 IC50 = 6600 nM T78429 CJ7H9M 52942943 IC50 = 42 nM T78429 C6OTY5 53251320 IC50 = 24000 nM T78429 CA03JM 53252601 IC50 = 900 nM T78429 CTIG48 53252602 IC50 = 200 nM T78429 C32TCY 53252779 IC50 = 2300 nM T78429 CT43EM 53252870 IC50 = 4500 nM T78429 CHEF79 53316855 IC50 = 71 nM T78429 C2U6FN 53316856 IC50 = 22 nM T78429 CBW02V 53316857 IC50 = 7300 nM T78429 CWG0U2 53316873 IC50 = 3.5 nM T78429 C56TPI 53316874 IC50 = 10 nM T78429 C0LV3O 53316875 IC50 = 7.6 nM T78429 CSG5M8 53316876 IC50 = 2.8 nM T78429 CXS83V 53316877 IC50 = 1.1 nM T78429 C47LNY 53316878 IC50 = 2.5 nM T78429 CFY6E5 53316879 IC50 = 10.2 nM T78429 C3W5EP 53317261 IC50 = 41 nM T78429 C5QCR2 53317336 IC50 = 500 nM T78429 CRC13Q 53317640 IC50 = 12 nM T78429 CE8OY2 53317913 IC50 > 100 nM T78429 CW5K8X 53318177 IC50 = 97 nM T78429 CNL25X 53318191 IC50 = 2.8 nM T78429 C9ERV1 53318192 IC50 = 4.2 nM T78429 CG86PO 53318194 IC50 = 2.3 nM T78429 CJU9N2 53318547 IC50 = 49 nM T78429 CFZN31 53318915 IC50 = 2900 nM T78429 C9KZB8 53318974 IC50 = 3.5 nM T78429 CVG50H 53319529 IC50 = 13 nM T78429 C6ZBL2 53319540 IC50 = 1.2 nM T78429 C2Y1UB 53319541 IC50 = 14 nM T78429 CTK9X2 53319542 IC50 = 4.3 nM T78429 C0WIU8 53319545 IC50 = 6.6 nM T78429 C0QON9 53319546 IC50 = 1.4 nM T78429 CY6Z9A 53319547 IC50 = 1 nM T78429 C3QWU5 53319869 IC50 = 34 nM T78429 C0GID9 53319942 IC50 = 2200 nM T78429 CQST54 53319943 IC50 = 3100 nM T78429 CPY2E5 53320356 IC50 = 0.5 nM T78429 C64CEL 53320812 IC50 = 23 nM T78429 CU09MT 53320813 IC50 = 15 nM T78429 C3MPK9 53320832 IC50 = 2.2 nM T78429 CMGT59 53320833 IC50 = 3.9 nM T78429 CX5G6M 53321170 IC50 = 60 nM T78429 C29PES 53321171 IC50 = 55 nM T78429 C3CN5V 53321172 IC50 = 36 nM T78429 C9ODE4 53321173 IC50 = 39 nM T78429 C6Q1NG 53321174 IC50 = 20 nM T78429 C6U7ON 53321244 IC50 = 8400 nM T78429 CJ69MU 53321245 IC50 = 7100 nM T78429 CA21YD 53321246 IC50 = 4800 nM T78429 C8H3LE 53321247 IC50 > 10000 nM T78429 CV1T5R 53321248 IC50 = 2500 nM T78429 C1O4MK 53321249 IC50 = 1900 nM T78429 CCRQ48 53321250 IC50 > 10000 nM T78429 C52ZJQ 53321634 IC50 = 17 nM T78429 C5L1TJ 53321705 IC50 > 500 nM T78429 C9FL4Y 53322167 IC50 = 3 nM T78429 CV5FA0 53322168 IC50 = 3.7 nM T78429 C8TYM9 53322169 IC50 = 1.3 nM T78429 C9PR6L 53322170 IC50 = 0.9 nM T78429 CLUS24 53322171 IC50 = 3.3 nM T78429 CX7F2G 53322492 IC50 = 57 nM T78429 CQZN03 53322493 IC50 = 130 nM T78429 CR92LT 53322494 IC50 = 78 nM T78429 CWNI81 53322965 IC50 = 110 nM T78429 C23WYK 53323485 IC50 = 17 nM T78429 C17DNC 53323502 IC50 = 2.8 nM T78429 C80FVL 53323503 IC50 = 6.1 nM T78429 CG0QH5 53323504 IC50 = 0.6 nM T78429 C0E2WG 53323505 IC50 = 5 nM T78429 C6QOL1 53323840 IC50 = 27 nM T78429 C6IS2B 53323910 IC50 = 500 nM T78429 C4NS7U 53324277 IC50 = 4.7 nM T78429 C6QCJ3 53324309 IC50 = 18 nM T78429 CIAS02 53324796 IC50 = 42 nM T78429 CC1K9J 53324797 IC50 = 15 nM T78429 C2A3JB 53324815 IC50 = 0.6 nM T78429 C7HQD2 53324816 IC50 = 14 nM T78429 C4CD0I 53324817 IC50 = 1 nM T78429 CM6J4E 53324818 IC50 = 2.2 nM T78429 CR8HQ3 53324819 IC50 = 0.5 nM T78429 C5Q6IG 53325111 IC50 = 16 nM T78429 C6UH5Q 53325112 IC50 = 10 nM T78429 CUG3D4 53325187 IC50 = 2200 nM T78429 CC4UA6 53325560 IC50 = 100 nM T78429 CSF3V9 53325628 IC50 = 21 nM T78429 CCZ53L 53326095 IC50 = 4.8 nM T78429 C94XDW 53326096 IC50 = 1.9 nM T78429 CQ6F9H 53326097 IC50 = 2 nM T78429 CXDJ40 53326098 IC50 = 1.3 nM T78429 C12CLZ 53326416 IC50 = 28 nM T78429 C4SKU0 53326482 IC50 = 8800 nM T78429 C2DQM0 53326483 IC50 = 900 nM T78429 C8ZRE3 53356518 IC50 > 50000 nM T78429 CB57NE 53363921 IC50 = 17 nM T78429 C8NA4L 53384644 IC50 > 30000 nM T78429 CGB86L 54580034 IC50 = 3800 nM T78429 CIK9F2 54580282 IC50 = 1258.93 nM T78429 CRF0L1 54581026 IC50 = 3670 nM T78429 C8R0GT 54581284 IC50 = 794.33 nM T78429 CX6BG5 54581285 IC50 > 15848.93 nM T78429 C51JPF 54582174 IC50 = 2200 nM T78429 C5V6OY 54582175 IC50 = 1300 nM T78429 CC46XA 54582474 IC50 > 15848.93 nM T78429 CDT9Q6 54583140 IC50 = 19700 nM T78429 C0CVM2 54583141 IC50 = 7020 nM T78429 CF62LG 54584009 IC50 = 3200 nM T78429 CI7Y3B 54585061 IC50 = 2090 nM T78429 CF5TS9 54585210 IC50 = 6309.57 nM T78429 CNUP53 54586040 IC50 = 920 nM T78429 C5N6EG 54586041 IC50 = 5600 nM T78429 C53JWF 54587018 IC50 = 4250 nM T78429 CVS2F1 54587019 IC50 = 3140 nM T78429 CSP4Y0 54587020 IC50 = 3850 nM T78429 CE2XK3 54587170 IC50 = 1584.89 nM T78429 CE1ZK6 54759168 IC50 > 10000 nM T78429 C9EMO2 54765177 IC50 = 288 nM T78429 CN9QD7 56643097 IC50 > 10000 nM T78429 CEDB74 56659739 IC50 = 300 nM T78429 CPA63X 56659740 IC50 = 43 nM T78429 C5X0DI 56659881 IC50 = 6300 nM T78429 CA3J0N 56663214 IC50 = 64 nM T78429 C6BPQ0 56663215 IC50 = 140 nM T78429 CX5O0H 56663216 IC50 = 19000 nM T78429 CZN15M 56663217 IC50 = 64 nM T78429 C5U2CL 56663218 IC50 = 19 nM T78429 CH7W6S 56663340 IC50 = 710 nM T78429 CY48RS 56663342 IC50 = 620 nM T78429 C0NQ4Y 56666651 IC50 = 71 nM T78429 CDE85V 56666652 IC50 = 27 nM T78429 CA5B6P 56666653 IC50 = 16 nM T78429 CIGH81 56666772 IC50 = 200 nM T78429 CO31CQ 56666813 IC50 = 8 nM T78429 CYE8H0 56670065 IC50 = 26 nM T78429 C4FHR6 56670204 IC50 = 1600 nM T78429 C5CSV7 56670206 IC50 = 420 nM T78429 CB1TG8 56670207 IC50 = 964 nM T78429 CZ74CL 56673590 IC50 = 410 nM T78429 CE7X6P 56673591 IC50 = 200 nM T78429 CP2EI4 56673592 IC50 = 29 nM T78429 CCF98O 56673729 IC50 = 300 nM T78429 CBFS82 56676913 IC50 = 680 nM T78429 CZ6D7V 56676914 IC50 = 120 nM T78429 C6C3ZA 56677035 IC50 = 12700 nM T78429 C3UV6G 56680221 IC50 = 97 nM T78429 CK6GV4 56680222 IC50 = 61 nM T78429 C3K5JV 56680361 IC50 = 980 nM T78429 C0ZB7X 56680362 IC50 = 273 nM T78429 CABX36 56683563 IC50 = 140 nM T78429 CAL69G 56683693 IC50 = 560 nM T78429 C9W5HU 56683694 IC50 = 331 nM T78429 CT4E8R 56832546 IC50 = 34000 nM T78429 CBOD63 56835089 IC50 > 30000 nM T78429 CX75NT 57390441 IC50 = 8170 nM T78429 CGN9C6 57391444 IC50 = 19 nM T78429 C87YVO 57391445 IC50 = 9 nM T78429 CD5OZ3 57391446 IC50 = 44 nM T78429 CV80UG 57391447 IC50 = 28 nM T78429 CP4JN3 57391448 IC50 = 20 nM T78429 CXRN14 57392233 IC50 = 13140 nM T78429 CZ7R5A 57393212 IC50 = 81 nM T78429 C20RWG 57393213 IC50 = 33 nM T78429 C79IBT 57393214 IC50 = 12 nM T78429 CC2PL8 57393215 IC50 = 5 nM T78429 C7QUM8 57393216 IC50 = 19 nM T78429 CVY21E 57393217 IC50 = 128 nM T78429 CD97JC 57393978 IC50 = 6600 nM T78429 CL0X9R 57393979 IC50 = 41650 nM T78429 CU3WD7 57394932 IC50 = 14 nM T78429 C7SXV0 57394933 IC50 = 23 nM T78429 CH76BE 57394934 IC50 = 12 nM T78429 CF2Z3E 57394935 IC50 = 130 nM T78429 CIWG72 57394936 IC50 = 438 nM T78429 CD6Y9Z 57395116 IC50 > 30000 nM T78429 C8W6IG 57395117 IC50 > 30000 nM T78429 C7P5BW 57395741 IC50 = 25300 nM T78429 CZ2XA5 57396689 IC50 = 330 nM T78429 CG7S0D 57396882 IC50 > 30000 nM T78429 CE6JK4 57398455 IC50 = 66 nM T78429 C0TV5O 57398456 IC50 = 41 nM T78429 C4V1JH 57399200 IC50 = 40270 nM T78429 CU9W3I 57400123 IC50 = 86 nM T78429 C21EVI 57400963 IC50 = 10780 nM T78429 C0UDY9 57401151 IC50 > 30000 nM T78429 C1PF3A 57402010 IC50 = 5.7 nM T78429 C0UAD3 57403655 IC50 = 26 nM T78429 CI6TF1 57403656 IC50 = 13 nM T78429 C7MS8X 57446795 IC50 = 53000 nM T78429 C8R4FE 57991377 IC50 = 375.4 nM T78429 CB82IK 58801625 IC50 = 28.18 nM T78429 C6BPR2 58985201 IC50 > 30000 nM T78429 CNV56K 59332591 IC50 = 7.943 nM T78429 CS14RJ 59332600 IC50 = 7.943 nM T78429 C5E3CW 59332772 IC50 = 158.49 nM T78429 C1WJD3 59406184 IC50 = 79.43 nM T78429 CS8F3Q 59406262 IC50 = 794.33 nM T78429 CVY3C8 59406271 IC50 = 12.59 nM T78429 CXJ63M 59603829 IC50 > 100000 nM T78429 CQEU96 59603842 IC50 > 10000 nM T78429 CSPD01 59744353 IC50 = 7.943 nM T78429 CC8T7R 59744382 IC50 = 6.31 nM T78429 CM1S2I 59744412 IC50 = 19.95 nM T78429 C0SBK4 59744417 IC50 = 7.943 nM T78429 C6PB3C 59744422 IC50 = 5.012 nM T78429 C7JDY6 59744451 IC50 = 6.31 nM T78429 C8Q2MN 59744508 IC50 = 3.981 nM T78429 C56DCI 59744533 IC50 = 19.95 nM T78429 CMB8X7 59744546 IC50 = 15.85 nM T78429 C23NOS 59744560 IC50 = 7.943 nM T78429 C4QLN7 59744593 IC50 = 15.85 nM T78429 C3M6SK 59828969 IC50 = 79.43 nM T78429 C1MR8Q 60097495 IC50 > 10000 nM T78429 CL36SQ 61992242 IC50 > 100000 nM T78429 CNP85L 61992815 IC50 = 50900 nM T78429 CU28AB 62900145 IC50 > 100000 nM T78429 CHKM07 66554457 IC50 = 10700 nM T78429 CI7WB0 66745713 IC50 = 100 nM T78429 CZ5H8O 66746880 IC50 = 39.81 nM T78429 CV63UL 67240318 IC50 > 10000 nM T78429 CWU52N 68790681 IC50 = 19.95 nM T78429 CU8G2Y 68792332 IC50 = 190 nM T78429 C9AC1O 68794144 IC50 = 6.31 nM T78429 C5DGR9 69036886 IC50 = 10000 nM T78429 C3GTU1 69762142 IC50 > 10000 nM T78429 CRO28P 70682547 IC50 = 8500 nM T78429 COZ28E 70682548 IC50 = 4200 nM T78429 C6OC1U 70684631 IC50 = 6300 nM T78429 CY2KE0 70684634 IC50 = 2600 nM T78429 CC9M8P 70686777 IC50 = 7300 nM T78429 C8NVG0 70686778 IC50 = 5700 nM T78429 CIR17F 70688862 IC50 = 14100 nM T78429 CQ8HE2 70690944 IC50 = 350 nM T78429 C17BKZ 70693089 IC50 = 230 nM T78429 C4AL6D 70693090 IC50 = 8700 nM T78429 C13FWG 70695135 IC50 = 1500 nM T78429 C1MUT2 70695137 IC50 = 6300 nM T78429 C1NJ4O 70695139 IC50 = 23600 nM T78429 C2OU9J 70697172 IC50 = 3300 nM T78429 C0VZB2 70697173 IC50 = 1500 nM T78429 C8HJQ1 70697174 IC50 = 160 nM T78429 CFD5R6 70697175 IC50 = 15600 nM T78429 CXO6A9 70697177 IC50 = 9300 nM T78429 CH0B8N 70789756 IC50 > 30000 nM T78429 CQ31PG 71138120 Ki > 30000 nM T78429 C91HPI 71300299 IC50 > 5000 nM T78429 CEBO91 71452977 IC50 > 10000 nM T78429 CHQZ25 71459584 IC50 > 10000 nM T78429 CA2V1U 71462267 IC50 = 15.85 nM T78429 CCN01X 71547862 IC50 > 10000 nM T78429 CA3O6K 71552696 IC50 = 17260 nM T78429 C1NPL0 71552941 IC50 > 30000 nM T78429 CA4PS8 71552942 IC50 > 30000 nM T78429 C3UA9C 71553011 IC50 = 30000 nM T78429 CEZ15Y 71553012 IC50 = 30000 nM T78429 CVIA91 71553085 IC50 = 30000 nM T78429 C1TR3O 71553152 IC50 = 30000 nM T78429 CZ31PU 71583657 IC50 > 10000 nM T78429 CP1DI5 71655874 IC50 = 790 nM T78429 C9DGO1 71655906 IC50 = 820 nM T78429 C3AUT6 71656001 IC50 = 2100 nM T78429 CA0QD7 71656003 IC50 = 600 nM T78429 C7UDL9 71656005 IC50 = 640 nM T78429 C1SKB0 71656007 IC50 = 840 nM T78429 CBM8Q7 71656015 IC50 = 1130 nM T78429 CN38TU 71656021 IC50 = 900 nM T78429 C4HTK1 71656031 IC50 = 790 nM T78429 CVC61J 71699285 IC50 = 4240 nM T78429 CXSI14 71718330 IC50 = 15000 nM T78429 C1TM3P 71720141 IC50 = 15000 nM T78429 C2XZW3 72708899 IC50 > 40000 nM T78429 CKN46T 72708901 IC50 > 40000 nM T78429 CRLG23 73345800 IC50 = 15.14 nM T78429 CF8I3C 73345801 IC50 = 2511.89 nM T78429 COD3J9 73345802 IC50 = 25.7 nM T78429 C43EHW 73346049 IC50 = 2620 nM T78429 CB03AU 73347278 IC50 = 15.14 nM T78429 C7Y6OZ 73348798 IC50 = 446.68 nM T78429 C94BXR 73350370 IC50 = 39.81 nM T78429 C9L6QE 73351880 IC50 = 100000 nM T78429 CRI4Y1 73351886 IC50 > 100000 nM T78429 C6IE8X 73353353 IC50 = 100000 nM T78429 C8MPS5 73354864 IC50 = 33.11 nM T78429 CV1UC7 73354865 IC50 = 316.23 nM T78429 CG29VX 73354866 IC50 = 15848.93 nM T78429 C6F9GQ 73354867 IC50 = 10000 nM T78429 CDB0Q6 73354870 IC50 = 15.14 nM T78429 CF6AV2 73354871 IC50 = 229.09 nM T78429 CA2WL9 73356420 IC50 = 117.49 nM T78429 CX4GU7 76317752 IC50 = 940 nM T78429 C19WQM 76321443 IC50 = 5160 nM T78429 CDB32S 76321457 IC50 = 1200 nM T78429 C93APE 76325038 IC50 = 4430 nM T78429 CB04OD 82482456 IC50 > 100000 nM T78429 C1HW4B 89735655 IC50 = 31000 nM T78429 CK6V9J 90644118 IC50 > 50000 nM T78429 CY0UC4 90645194 IC50 > 10000 nM T78429 CAU45T 91971978 IC50 > 30000 nM T78429 CXU1Z2 101043725 IC50 = 14 nM T78429 C75AVW 102334651 Ki = 3600 nM T78429 CM9Y8O 117073666 IC50 = 41000 nM T78429 CY7BI2 118706214 IC50 > 10000 nM T78429 C3T1DS 118708699 IC50 = 1360 nM T78429 CE59BN 118708701 IC50 = 1540 nM T78429 CQCX41 118737057 IC50 = 164 nM T78429 CLX5Y9 127026219 IC50 = 9880 nM T78429 CQ7P0J 127026816 IC50 = 960 nM T78429 CN23QK 127032120 IC50 = 579 nM T78429 CNP5O7 127033734 IC50 = 324 nM T78429 C1R4HV 127033748 IC50 = 773 nM T78429 CHIQ36 127040246 IC50 = 850 nM T78429 CZ5B8J 127040247 IC50 = 840 nM T78429 CC29FJ 127040248 IC50 = 820 nM T78429 C0EJS9 129320519 Ki = 2300 nM T78429 CJE3H1 134130251 IC50 = 111000 nM T78429 CW5TF4 134130801 IC50 > 20000 nM T78429 C6IBY4 134132116 IC50 = 8100 nM T78429 C15IHV 134134683 IC50 = 1100 nM T78429 C24FMI 134135188 IC50 = 65000 nM T78429 CKOY19 134138404 IC50 = 1600 nM T78429 CN07WL 134138531 IC50 > 50000 nM T78429 C6NV9O 134138868 IC50 = 4600 nM T78429 CE06AV 134140298 IC50 = 14200 nM T78429 C7ONY0 134141927 IC50 = 34 nM T78429 C69BYF 134143911 IC50 = 11800 nM T78429 CW5QJ3 134144073 IC50 = 320 nM T78429 CJ65ZO 134145999 IC50 = 2700 nM T78429 C06NPQ 134146120 IC50 = 28700 nM T78429 CK2PN1 134146398 IC50 = 97 nM T78429 CYXM38 134147237 IC50 = 4200 nM T78429 CJR26T 134148194 IC50 = 1100 nM T78429 C03TLW 134149798 IC50 = 190000 nM T78429 C8XVB7 134149926 IC50 = 79000 nM T78429 C9DK1I 134150942 IC50 = 138000 nM T78429 CPI16E 134152111 IC50 = 6200 nM T78429 CV75DE 134153774 IC50 = 1520 nM T78429 C5WYO4 134154113 IC50 = 34100 nM T78429 C0TEL2 134155081 IC50 = 12000 nM T78429 CN64UH 134156138 IC50 > 20000 nM T78429 C2AN7T 134611886 IC50 > 100000 nM T78429 C54FXD 134957362 IC50 > 10000 nM T78429 CKHV90 135401952 IC50 = 7943.28 nM T78429 CB29GK 135403018 IC50 = 670 nM T78429 CZ07HB 135427928 IC50 = 316 nM T78429 CD8V9X 135432858 IC50 = 25 nM T78429 CQX0Z6 135443473 IC50 = 12 nM T78429 CEP9R5 135443474 IC50 = 3.981 nM T78429 COV4L9 135454904 Ki = 2 nM T78429 CRY3K8 135456003 IC50 = 600 nM T78429 CJ3F0V 135458385 IC50 = 3 nM T78429 C2OH3D 135462238 IC50 = 19952.62 nM T78429 CQM48T 135468292 IC50 > 15500 nM T78429 CUGI96 135469484 IC50 = 9.12 nM T78429 C86WCU 135469510 IC50 = 1500 nM T78429 CQAJ91 135469553 IC50 = 600 nM T78429 CY63WC 135482239 IC50 = 5 nM T78429 CV49XC 135484475 IC50 = 24 nM T78429 C2QB1M 135495606 IC50 = 10800 nM T78429 C5YC4F 135495607 IC50 = 6980 nM T78429 CW0S3I 135513122 IC50 = 120 nM T78429 C56WYX 135527124 IC50 = 25 nM T78429 C3GSZ2 135529859 IC50 = 19952.62 nM T78429 C9I8TR 135530494 IC50 = 500 nM T78429 CKCI43 135543029 IC50 = 800 nM T78429 C70MNK 135550601 IC50 = 230 nM T78429 CC9AT3 135550610 IC50 = 7800 nM T78429 CEK31P 135566415 IC50 > 20000 nM T78429 CV68FG 135584950 IC50 = 40 nM T78429 CIA1O9 135584951 IC50 = 80 nM T78429 C7GR1F 135584952 IC50 = 240 nM T78429 CC8D6V 135584953 IC50 = 60 nM T78429 CVYA94 135584954 IC50 = 730 nM T78429 CGVC82 135584955 IC50 = 150 nM T78429 CZEP45 135584956 IC50 = 480 nM T78429 C6YJ3N 135584957 IC50 = 110 nM T78429 C4DI5N 135584958 IC50 = 70 nM T78429 CJ7XQ9 135584959 IC50 = 470 nM T78429 C28WOL 135584961 IC50 = 15 nM T78429 CT4BN0 135584962 IC50 = 270 nM T78429 CAUR52 135584963 IC50 = 110 nM T78429 C5IHB8 135584964 IC50 = 15.14 nM T78429 CX9DJ1 135584965 IC50 = 26 nM T78429 C0IUF3 135584967 IC50 = 14 nM T78429 CB57KR 135584968 IC50 = 14 nM T78429 CMR9C1 135584969 IC50 = 50 nM T78429 C3PHM9 135584970 IC50 = 1300 nM T78429 CDT1V6 135584971 IC50 = 5 nM T78429 C73ASO 135584972 IC50 = 15 nM T78429 C4DMJ3 135584973 IC50 = 81 nM T78429 CE23GS 135584974 IC50 = 33.88 nM T78429 C8LCS3 135584975 IC50 = 2400 nM T78429 C3L5QR 135584976 IC50 = 6 nM T78429 C2D6WL 135584977 IC50 = 19.95 nM T78429 C2YG7L 135584978 IC50 = 230 nM T78429 CG5FM3 135584980 IC50 = 530 nM T78429 CP4C0V 135584981 IC50 = 300 nM T78429 C9V0HX 135584984 IC50 = 6500 nM T78429 CXM86H 135584989 IC50 = 330 nM T78429 CX4ZB3 135863110 IC50 > 10000 nM T78429 CV24UR 135873213 IC50 = 10000 nM T78429 CV76UY 135909516 IC50 > 15848.93 nM T78429 CHA4N2 136013680 IC50 > 10 nM T78429 CC9X6K 136053669 IC50 = 6200 nM T78429 CPQ0G6 136053670 IC50 = 20000 nM T78429 CI7MS9 136053671 IC50 = 560 nM T78429 C7GQX6 136059717 IC50 = 8 nM T78429 CK30FD 136078537 IC50 > 20000 nM T78429 C1KT0O 136078539 IC50 = 500 nM T78429 C3S4JG 136078541 IC50 = 600 nM T78429 C34TDM 136078542 IC50 = 600 nM T78429 C5V0CM 136078543 IC50 = 1400 nM T78429 CUWK81 136094897 IC50 = 1000 nM T78429 CD5AZ7 136094904 IC50 = 1000 nM T78429 CT5QM6 136094910 IC50 = 20000 nM T78429 COY84Z 136094911 IC50 > 20000 nM T78429 CNY64Q 136094913 IC50 = 2500 nM T78429 C8LIE3 136094916 IC50 = 1800 nM T78429 CSB1N0 136094917 IC50 = 3000 nM T78429 CVTX18 136094920 IC50 = 1400 nM T78429 C5HP8X 136094921 IC50 = 15000 nM T78429 C79CSM 136114625 IC50 = 700 nM T78429 CDI2P9 136114626 IC50 > 20000 nM T78429 CJX7D0 136114627 IC50 > 20000 nM T78429 C8YWE0 136114629 IC50 = 900 nM T78429 CN3S9C 136114630 IC50 = 2000 nM T78429 CG74JM 136114631 IC50 = 5500 nM T78429 CFZC45 136114632 IC50 = 1700 nM T78429 CTQX39 136114640 IC50 = 700 nM T78429 CFW6U4 136114641 IC50 = 2500 nM T78429 C9A8VY 136114642 IC50 = 5300 nM T78429 CK4MY5 136180744 IC50 > 20000 nM T78429 CZ7EX0 136183413 IC50 > 30000 nM T78429 C1YUD0 136219394 IC50 > 10 nM T78429 CLG1Y2 136224215 IC50 = 7810 nM T78429 CAF61N 136249387 IC50 = 4780 nM T78429 CIU8W3 136254389 IC50 > 10 nM T78429 CW36RX 136254398 IC50 = 8.511 nM T78429 CB32UM 136264284 IC50 = 3370 nM T78429 CR83YE 137631544 Ki > 30000 nM T78429 CT0P5R 137632102 Ki > 30000 nM T78429 C5CU9T 137632103 Ki = 20000 nM T78429 C6FJ1P 137632317 Ki = 5900 nM T78429 CB9XT2 137632532 Ki = 2500 nM T78429 C6W2PJ 137633160 Ki = 100 nM T78429 CDBV08 137634477 Ki > 30000 nM T78429 C0KU4C 137635130 Ki > 30000 nM T78429 C8F7OK 137636751 Ki > 30000 nM T78429 CVZ5Y6 137637765 Ki = 300 nM T78429 CK08TL 137640054 Ki > 30000 nM T78429 C3FNV9 137640501 Ki > 30000 nM T78429 C8BF9I 137640852 Ki > 30000 nM T78429 C02MPZ 137641352 Ki = 400 nM T78429 C2L6ZU 137641677 Ki = 1000 nM T78429 C1Y6NI 137641784 Ki > 30000 nM T78429 C7BQX5 137642493 Ki > 30000 nM T78429 CSZ6B9 137643197 Ki > 30000 nM T78429 CC0T7J 137644890 Ki > 30000 nM T78429 C2QSP4 137645617 Ki > 30000 nM T78429 CS9T4Q 137646916 Ki > 30000 nM T78429 C5P2NR 137648275 Ki > 30000 nM T78429 CA84NC 137648771 Ki > 30000 nM T78429 CH2S7I 137648911 Ki > 30000 nM T78429 C5QMA7 137648912 Ki > 30000 nM T78429 C2AN5P 137650396 Ki = 5900 nM T78429 CKW51R 137650911 Ki > 30000 nM T78429 C6VHT8 137651289 Ki > 30000 nM T78429 CS9WT0 137651927 Ki > 30000 nM T78429 C6L5KV 137652726 Ki > 30000 nM T78429 CZ1L7Y 137653022 Ki = 3800 nM T78429 C1G3KP 137653092 Ki > 30000 nM T78429 CP5X0N 137653110 Ki > 30000 nM T78429 C5TJ8K 137653144 Ki = 4000 nM T78429 C9AIU6 137655282 Ki = 610 nM T78429 C0M4KH 137655668 Ki > 30000 nM T78429 CGKU15 137655801 Ki > 30000 nM T78429 CE8N2X 137655941 Ki > 30000 nM T78429 CGW9I0 137656387 IC50 = 6230 nM T78429 CYKL36 137656635 Ki > 30000 nM T78429 CF41YQ 137656752 Ki > 30000 nM T78429 C86SIX 137657214 Ki > 30000 nM T78429 C3VT5X 137657569 Ki > 30000 nM T78429 CA7RD3 137657800 Ki = 20000 nM T78429 C7S2EH 137657801 Ki > 30000 nM T78429 COXH36 137659346 Ki = 1400 nM T78429 C2BRJ0 137659655 Ki > 30000 nM T78429 CCNA02 137660360 Ki > 30000 nM T78429 COS48M 137661213 Ki > 30000 nM T78429 C9O3EJ 137661645 Ki > 30000 nM T78429 CLBV34 137661772 Ki > 30000 nM T78429 C6VB3O 145925651 IC50 >= 5000 nM T78429 CT89FP 145952913 IC50 > 100000 nM T78429 C1E6MX 145957558 IC50 = 14000 nM T78429 CDNC31 145967951 IC50 > 500 nM T78429 C91BHP 145971744 IC50 = 1720 nM T78429 CML8O0 145979124 IC50 > 100000 nM T78429 CVJO79 145979309 IC50 = 97400 nM T78429 CK20XI 145979715 IC50 > 200000 nM T78429 CQLH68 145979774 IC50 > 100000 nM T78429 C5YR8W 145979893 IC50 > 100000 nM T78429 CGL48D 145980076 IC50 > 100000 nM T78429 C5LK9A 145980083 IC50 > 100000 nM T78429 CCSY15 145980681 IC50 > 100000 nM T78429 CSEC23 145980764 IC50 = 1500 nM T78429 CY80PH 145981483 IC50 > 100000 nM T78429 CN3U5W 145981500 IC50 > 100000 nM T78429 CFSQ94 145981688 IC50 > 100000 nM T78429 CI3P2B 145981824 IC50 = 25900 nM T78429 CK1WG0 145982087 IC50 > 200000 nM T78429 C1BP0G 145982116 IC50 = 7900 nM T78429 CW89QD 145984138 IC50 = 900 nM T78429 CVRZ23 145984375 IC50 > 100000 nM T78429 CH7GD5 145986473 IC50 > 200000 nM T78429 CGE7B8 145987124 IC50 > 100000 nM T78429 C86HGI 145987159 IC50 > 100000 nM T78429 CU3J8R 145987461 IC50 > 100000 nM T78429 C59OKW 145987584 IC50 = 8600 nM T78429 CW7V1O 145987719 IC50 > 2000 nM T78429 CRJQ18 145988918 IC50 > 100000 nM T78429 C8QH2W 145989390 IC50 = 22900 nM T78429 CFAK86 145989643 IC50 > 100000 nM T78429 CHWR01 145989760 IC50 = 1320 nM T78429 C3EIA1 145990026 IC50 > 100000 nM T78429 CBZ94U 145990465 IC50 > 100000 nM T78429 C8M5AU 145990524 IC50 > 100000 nM T78429 C4FQ0C 145990918 IC50 > 100000 nM T78429 CN38UG 145990988 IC50 > 100000 nM T78429 CGSZ75 145991182 IC50 > 100000 nM T78429 C2SY4M 145991367 IC50 = 6930 nM T78429 C0CJ9I 145991401 IC50 = 42800 nM T78429 CI60XK 145991710 IC50 = 143 nM T78429 C17TOS 145991715 IC50 > 100000 nM T78429 C68ZYI 145991820 IC50 = 90 nM T78429 C9YWM0 145991838 IC50 = 1700 nM T78429 C3HIB8 145992014 IC50 > 100000 nM T78429 CMN54B 145992036 IC50 = 68000 nM T78429 CF28WP 145992122 IC50 > 100000 nM T78429 C85OWM 145992355 IC50 > 100000 nM T78429 C50OJM 145992513 IC50 = 252.35 nM T78429 CD54KY 145992596 IC50 > 100000 nM T78429 CJC20Z 145992663 IC50 = 1400 nM T78429 CQI81V 145992947 IC50 = 13600 nM T78429 CQ8V6K 145993087 IC50 > 200000 nM T78429 C3NU7C 145993088 IC50 > 100000 nM T78429 CIVT98 145993430 IC50 = 400 nM T78429 C0CJ9B 145993626 IC50 = 47700 nM T78429 C2GH5C 145993662 IC50 > 100000 nM T78429 CMJ6G4 145993951 IC50 > 100000 nM T78429 CA06KI 145994056 IC50 = 71300 nM T78429 CY27DC 155511489 IC50 = 125.89 nM T78429 C2MD1Q 155513187 IC50 > 10000 nM T78429 C5YKT4 155520282 IC50 = 501.19 nM T78429 C35OXY 155521834 IC50 = 39.81 nM T78429 C2CG1A 155537016 IC50 > 10000 nM T78429 CHAY47 155550017 IC50 = 79.43 nM T78429 CA8ZV0 155550321 IC50 = 63.1 nM T78429 C8HX3K 155554640 IC50 = 19.95 nM T78429 CTL4A2 155555619 IC50 = 501.19 nM T78429 CSHT68 155555784 IC50 = 199.53 nM T78429 D00ERW 44444843 Ki > 2338 nM T78429 D00HVA 11624601 Ki > 3200 nM T78429 D00XDG 11708263 IC50 = 11000 nM T78429 D00YTQ 9926054 IC50 = 300 nM T78429 D01FPX 11543063 IC50 = 12700 nM T78429 D03DZO 11715767 IC50 > 10000 nM T78429 D03MUZ 17759555 IC50 = 73000 nM T78429 D03OKV 9844320 IC50 > 10000 nM T78429 D03PVS 821974 IC50 = 12600 nM T78429 D04PEI 11467730 IC50 > 50000 nM T78429 D06CBR 703965 IC50 = 1900 nM T78429 D06WGX 9549184 IC50 > 25000 nM T78429 D07ADX 54764565 IC50 = 257 nM T78429 D07MQC 9949093 IC50 = 186 nM T78429 D08HFG 24809764 IC50 = 3800 nM T78429 D08VQM 2756390 IC50 = 6600 nM T78429 D09HVH 135566652 IC50 > 10 nM T78429 D09PLJ 11499583 IC50 = 970 nM T78429 D0E0XV 9903786 IC50 = 18 nM T78429 D0EW9J 10389239 IC50 > 200000 nM T78429 D0F0VD 135465539 IC50 = 8.5 nM T78429 D0F8QJ 5281813 IC50 > 10000 nM T78429 D0IR6U 5494425 IC50 = 300 nM T78429 D0LE7J 58221375 IC50 > 100000 nM T78429 D0ME9B 46868971 IC50 > 10 nM T78429 D0N1UB 5200228 IC50 = 9600 nM T78429 D0O6OH 71553154 IC50 = 30000 nM T78429 D0O8TE 52915756 IC50 = 20000 nM T78429 D0Q3NG 11715520 Ki > 3200 nM T78429 D0S7IE 11658882 Ki > 3200 nM T78429 D0T6VA 2807869 IC50 = 1300 nM T78429 D0T8IS 9929127 IC50 = 465 nM T78429 D0UP6G 11600944 IC50 = 14500 nM T55729 D0EG1I 9926791 IC50 > 10000 nM T55729 D02NNV 3038525 Ki = 220 nM T55729 D0A1WN 11714580 IC50 = 23 nM T55729 D0C8DD 11552706 Ki = 25.12 nM T55729 D0K2ZF 22049997 Ki = 40 nM T55729 D0O6ZO 9952773 IC50 = 200 nM T55729 D0Q0AP 10409068 IC50 = 62 nM T55729 D0Q9UX 16718576 IC50 > 10000 nM T55729 D0F8DL 176155 IC50 = 12 nM T55729 D0T3ME 156422 IC50 = 7 nM T55729 C0SLP9 1489193 IC50 = 6309.57 nM T55729 C86LNP 2779952 IC50 > 100000 nM T55729 CL5I2U 5330279 IC50 > 10000 nM T55729 CQ57EC 9548013 IC50 > 100000 nM T55729 C20RSC 9811100 IC50 = 572 nM T55729 C4Z2GW 9819930 IC50 = 2408 nM T55729 C2L3NR 9826344 IC50 = 73 nM T55729 CQ3T8A 9827288 IC50 = 2540 nM T55729 CKG9P8 9844525 IC50 = 9780 nM T55729 CQH58C 9844883 IC50 = 4100 nM T55729 CDR82H 9865587 IC50 = 3450 nM T55729 CWYF96 9884921 IC50 = 2320 nM T55729 CJ4QV2 9885993 IC50 = 8.1 nM T55729 C3V6WA 9930407 IC50 = 10 nM T55729 CHD79R 9969008 IC50 = 110 nM T55729 CQP98N 10002079 IC50 = 52 nM T55729 C7YD1X 10048045 IC50 = 19 nM T55729 CEHV91 10134493 IC50 = 15 nM T55729 C69DHW 10158652 Ki = 160 nM T55729 CW3AH9 10319451 IC50 = 3250 nM T55729 C03UPC 10366721 IC50 = 57 nM T55729 C91FSN 11188019 IC50 = 10 nM T55729 C2W5RC 11235063 IC50 < 100 nM T55729 C71PYD 11427975 IC50 = 1.5 nM T55729 CJC95A 11454205 IC50 = 22 nM T55729 C5B3XJ 11620410 IC50 > 40000 nM T55729 CHB3F2 11626055 IC50 = 326 nM T55729 CGX96V 11626927 IC50 < 15848.93 nM T55729 CJ9KN7 11683817 IC50 = 249 nM T55729 CU53MJ 11685293 IC50 = 0.25 nM T55729 CU0E8O 11690457 Ki > 10000 nM T55729 CB0AP2 11705863 Ki > 10000 nM T55729 CWM32N 11957412 IC50 = 20 nM T55729 C9TU1O 16046126 IC50 > 1000 nM T55729 CL67VN 16049878 IC50 = 15 nM T55729 CM1C7H 17423309 IC50 = 784 nM T55729 CC1E7R 21078798 Ki = 440 nM T55729 C7I9VO 21088983 Ki = 6 nM T55729 CK4L1Y 21914620 Ki = 158.49 nM T55729 CZF82E 21914667 Ki = 25.12 nM T55729 CH73AW 22037206 IC50 = 404 nM T55729 CD2H1Z 22037230 IC50 = 3130 nM T55729 CXTL58 22037368 IC50 = 3450 nM T55729 CC1LM5 22037370 IC50 = 164 nM T55729 CK69RD 22037400 IC50 = 1050 nM T55729 CC7I8U 22037479 IC50 = 510 nM T55729 C38GTD 22037512 IC50 = 2680 nM T55729 CN2XE5 22037660 IC50 = 2520 nM T55729 CG4JS7 22037702 IC50 = 3530 nM T55729 CQ2T8N 22066045 IC50 = 3710 nM T55729 C0UMW7 22262550 IC50 = 1680 nM T55729 CR2H9V 22262560 IC50 = 3770 nM T55729 CN76KY 22953580 IC50 = 6720 nM T55729 CIVA91 22953801 IC50 = 6720 nM T55729 C5NJD7 22953832 IC50 = 1960 nM T55729 C75DWA 23400208 IC50 = 12 nM T55729 C7TSR0 23647364 IC50 = 990 nM T55729 CY34HX 23647366 IC50 = 450 nM T55729 C7Z0LW 23647367 IC50 = 920 nM T55729 C8S9KH 23647368 IC50 = 450 nM T55729 COEA71 23647369 IC50 = 850 nM T55729 CLW83Z 23647372 IC50 = 135 nM T55729 C0PN6O 23647373 IC50 = 211 nM T55729 C0U7GT 23647374 IC50 = 600 nM T55729 C4EX0K 23647375 IC50 = 41 nM T55729 C9G0TU 23647376 IC50 = 29 nM T55729 CQP59Z 23647378 IC50 = 29 nM T55729 C5KEF4 23647379 IC50 = 2 nM T55729 C2IA1Y 24794468 IC50 = 270 nM T55729 C61KPI 24856363 Ki = 24 nM T55729 CY8L7E 24896769 IC50 > 10000 nM T55729 C4CWQ9 24985573 IC50 = 265 nM T55729 CA01UI 24985915 IC50 = 81 nM T55729 CVQS96 25052767 Ki = 2.5 nM T55729 CL0Z1F 25181502 Ki = 1.8 nM T55729 C6G2FS 44326041 IC50 = 250 nM T55729 CS8Y4I 44351755 IC50 = 1230 nM T55729 CZF21R 44351880 IC50 = 200 nM T55729 CIEM10 44351882 IC50 = 250 nM T55729 CMG81Z 44351899 IC50 = 220 nM T55729 CWV8P9 44351908 IC50 = 530 nM T55729 CSG20K 44351945 IC50 = 530 nM T55729 CIK46B 44351950 IC50 = 950 nM T55729 CMJ9G4 44351956 IC50 = 2750 nM T55729 CUL6X2 44351971 IC50 = 190 nM T55729 CT4SH8 44351972 IC50 = 393 nM T55729 C7MHU6 44351974 IC50 = 980 nM T55729 CFL16M 44351990 IC50 = 1340 nM T55729 C5G7JS 44351997 IC50 = 800 nM T55729 CQZ5B8 44352051 IC50 = 1480 nM T55729 C5J0YM 44352052 IC50 = 2370 nM T55729 C47DES 44352068 IC50 = 220 nM T55729 CY6ST1 44352069 IC50 = 210 nM T55729 CLG9R7 44352098 IC50 = 3430 nM T55729 C6HN1F 44352102 IC50 = 52 nM T55729 CQG9P3 44352281 IC50 = 980 nM T55729 CXR91C 44419745 IC50 = 31 nM T55729 CU80BP 44517743 IC50 > 10000 nM T55729 C3VRO9 44557921 IC50 > 10000 nM T55729 C9VXN3 44578709 IC50 < 1000 nM T55729 CH3SF9 44631836 IC50 = 4 nM T55729 C61HBG 45102725 IC50 = 5400 nM T55729 C09BOA 46865979 IC50 = 3380 nM T55729 CYQ25D 46884595 IC50 = 3070 nM T55729 CXC97Z 46884596 IC50 = 2350 nM T55729 CS3UI6 46884597 IC50 = 3390 nM T55729 CY3T2E 46884634 IC50 = 6550 nM T55729 CQH28F 46884635 IC50 = 1650 nM T55729 CQ7E0D 46884636 IC50 = 4340 nM T55729 CIT8B5 46884665 IC50 = 1790 nM T55729 CT6Y1E 46884695 IC50 = 2780 nM T55729 C1EY3N 46884696 IC50 = 7410 nM T55729 CNH51B 46884697 IC50 = 9500 nM T55729 CC6BE5 46884730 IC50 = 3290 nM T55729 CET05C 46884779 IC50 = 3480 nM T55729 CJ97YS 49326850 IC50 = 18 nM T55729 CHSF07 49806372 IC50 > 1000 nM T55729 CEQN27 52936621 Ki > 1000 nM T55729 C8NA4L 53384644 IC50 = 50 nM T55729 C5V6OY 54582175 IC50 > 30000 nM T55729 CNUP53 54586040 IC50 = 210 nM T55729 CKA4M2 55786207 IC50 = 485 nM T55729 CS68PK 56659526 Ki = 17 nM T55729 C6UAN1 57467725 IC50 = 9714 nM T55729 C6VQ8S 58328161 IC50 = 7084 nM T55729 CYZ6X2 58328191 IC50 = 21920 nM T55729 C7WX9H 58328291 IC50 = 6173 nM T55729 C2JW1C 58328294 IC50 = 14890 nM T55729 C6BPR2 58985201 IC50 > 50000 nM T55729 C8MS1C 59749702 IC50 = 4 nM T55729 CL92GP 59761390 IC50 = 3875 nM T55729 CH21LA 59761399 IC50 = 1800 nM T55729 C5GAK1 59761424 IC50 = 332 nM T55729 C6DNV0 59761433 IC50 = 2402 nM T55729 CYV4E3 59761440 IC50 = 1021 nM T55729 CIO25V 59761450 IC50 = 771 nM T55729 CFSO82 59761454 IC50 = 6799 nM T55729 CIM3Z0 59761458 IC50 = 1514 nM T55729 C3MJC9 59761459 IC50 = 267 nM T55729 CRJ54F 59761462 IC50 = 390 nM T55729 CT51GX 59761498 IC50 = 679 nM T55729 CS41QF 59761509 IC50 = 441 nM T55729 CI3VU5 59761513 IC50 = 3455 nM T55729 C1MR8Q 60097495 IC50 > 10000 nM T55729 C26TWY 67148905 IC50 = 830 nM T55729 CV63UL 67240318 IC50 > 10000 nM T55729 CQ8HE2 70690944 IC50 > 30000 nM T55729 C13FWG 70695135 IC50 > 30000 nM T55729 C0VZB2 70697173 IC50 > 30000 nM T55729 C6ZW1R 71714236 IC50 = 492 nM T55729 CKV91X 71714379 IC50 = 109 nM T55729 CHC8Q5 71714380 IC50 = 254 nM T55729 CAI68B 71714533 IC50 = 409 nM T55729 C5GLM2 121232441 IC50 = 250 nM T55729 CGX6C4 136173253 IC50 = 36 nM T55729 CH2T5R 139030330 IC50 = 191 nM T55729 C7JEX9 139030331 IC50 = 144 nM T55729 COE1X5 139030332 IC50 = 550 nM T55729 CM3A8O 139030333 IC50 = 32 nM T55729 C42BWS 145994862 IC50 = 1600 nM T55729 CH9N0J 155511915 IC50 > 10000 nM T55729 CY1VF8 155511959 IC50 = 2970 nM T55729 CHEI63 155513115 IC50 > 10000 nM T55729 C2MD1Q 155513187 IC50 > 10000 nM T55729 C09TIS 155513203 IC50 = 5050 nM T55729 C4PDT6 155514077 IC50 = 370 nM T55729 CT5YG4 155514435 IC50 = 960 nM T55729 CWBU69 155514452 IC50 = 970 nM T55729 C6ZUK4 155514537 IC50 = 1960 nM T55729 C9O1QE 155515323 IC50 > 10000 nM T55729 CA54SV 155516886 IC50 = 99 nM T55729 CFG2M8 155517577 IC50 = 59 nM T55729 C0HZ8O 155518052 IC50 > 10000 nM T55729 CNE3Q5 155519237 IC50 > 10000 nM T55729 C68LNI 155519614 IC50 = 2180 nM T55729 C2YQ5I 155519636 IC50 > 10000 nM T55729 CUK59T 155520576 IC50 = 1160 nM T55729 CLH7Y2 155520781 IC50 = 3530 nM T55729 C6Z2QE 155522907 IC50 = 730 nM T55729 CM2QO4 155523988 IC50 > 10000 nM T55729 CYI5Z3 155524399 IC50 = 1700 nM T55729 CH95PJ 155524845 IC50 > 10000 nM T55729 C5E4WZ 155525348 IC50 > 10000 nM T55729 C3V8RW 155526111 IC50 = 2480 nM T55729 C2Z1AW 155526520 IC50 > 10000 nM T55729 CYQ1E0 155528481 IC50 > 10000 nM T55729 CQT70J 155529207 IC50 > 10000 nM T55729 CXFH38 155529296 IC50 = 167 nM T55729 CO2JD6 155529363 IC50 > 10000 nM T55729 C6ATZ2 155530054 IC50 > 10000 nM T55729 C58LZX 155531251 IC50 = 660 nM T55729 C0SR3H 155531653 IC50 > 10000 nM T55729 C48FKU 155533602 IC50 > 10000 nM T55729 CLZ32Q 155534860 IC50 = 4540 nM T55729 CMW7K0 155536680 IC50 = 6180 nM T55729 CQ39BV 155536797 IC50 = 209 nM T55729 CZ5A1P 155536847 IC50 > 10000 nM T55729 C24SFW 155537433 IC50 > 10000 nM T55729 CWP49G 155538536 IC50 > 10000 nM T55729 C6RD2N 155538801 IC50 > 10000 nM T55729 C46ICV 155539003 IC50 > 10000 nM T55729 C2S3FB 155542512 IC50 > 10000 nM T55729 CA5UN7 155542968 IC50 > 10000 nM T55729 CQ97ZD 155546227 IC50 > 10000 nM T55729 CC9LQ2 155546287 IC50 = 11000 nM T55729 C36BPF 155546292 IC50 = 328 nM T55729 C1FKM7 155546916 IC50 > 10000 nM T55729 CY96SD 155548355 IC50 > 10000 nM T55729 CW4LO3 155548563 IC50 = 3830 nM T55729 CT07RL 155548603 IC50 = 7050 nM T55729 C0X5EB 155549123 IC50 > 10000 nM T55729 CIQM72 155549185 IC50 > 10000 nM T55729 CB76ET 155549375 IC50 = 1282 nM T55729 CK9Z5W 155550010 IC50 > 10000 nM T55729 C26ILZ 155551090 IC50 = 736 nM T55729 CR0K3W 155551204 IC50 > 10000 nM T55729 CAQU49 155552777 IC50 > 10000 nM T55729 C7I9ER 155553064 IC50 > 10000 nM T55729 CDC59Q 155556256 IC50 = 1990 nM T55729 C1AIF0 155557307 IC50 = 7370 nM T55729 CND16A 155558659 IC50 > 10000 nM T55729 CPOV46 155560224 IC50 = 9890 nM T55729 CT39UJ 155561412 IC50 = 8700 nM T55729 C10FWR 155561550 IC50 = 4800 nM T55729 CUL57N 155562188 IC50 > 10000 nM T55729 CV1SK7 155563610 IC50 > 10000 nM T55729 C8N2FR 155564003 IC50 = 7300 nM T55729 C0P7QO 155565131 IC50 = 364 nM T55729 C5YXO3 155565855 IC50 > 10000 nM T55729 C4XT0Y 155565999 IC50 > 10000 nM T55729 CLA4I9 155566444 IC50 > 10000 nM T55729 CHZB01 155567574 IC50 > 10000 nM T55729 CLG3Y8 155568520 IC50 > 10000 nM T55729 C5P6AF 155568803 IC50 > 10000 nM T55729 D00NWF 5730 IC50 = 2000 nM T55729 D03DZO 11715767 IC50 > 10000 nM T55729 D04HWF 9871074 IC50 = 98 nM T55729 D08HFG 24809764 IC50 > 10000 nM T55729 D08LYB 5166 IC50 = 44 nM T55729 D0C7RS 1369 IC50 > 40000 nM T55729 D0QN6U 9806182 IC50 = 0.1 nM T55729 D0T8NU 16757525 IC50 > 4000 nM T55729 D0VC0I 5169 IC50 = 33.1 nM T23606 D0E3TC 44259 IC50 = 5.77 nM T23606 C2MD1Q 155513187 IC50 > 10000 nM T23606 D0N1UU 46871820 IC50 = 24 nM T96862 CJA29I 10382137 IC50 = 9 nM T96862 C0JX2B 44306130 IC50 = 150 nM T96862 CUH8V3 44306159 IC50 = 5000000 nM T96862 CR9XM6 44306161 IC50 = 300 nM T96862 D07GAU 44306132 Ki = 750 nM T96862 D0I0QH 44306087 Ki = 37 nM T02565 D00PEH 135449332 Ki = 25600 nM T02565 D00YZD 54726191 IC50 > 100000 nM T02565 D01TQR 72385 Ki = 2870 nM T02565 D02OZE 2724385 IC50 = 13182.57 nM T02565 D02RQU 54687 Ki = 57000 nM T02565 D02ZTJ 5339 Ki = 11000 nM T02565 D05VIX 3463 IC50 = 7079.46 nM T02565 D07IQS 148192 Ki = 370 nM T02565 D07POC 176870 Ki = 41000 nM T02565 D07UBG 130881 Ki = 750 nM T02565 D07VLY 31703 Ki = 38000 nM T02565 D09HNR 3002190 IC50 = 5888.44 nM T02565 D09QVV 5978 Ki = 9800 nM T02565 D0AZ8C 5213 Ki = 3270 nM T02565 D0B7EB 36462 IC50 = 4180 nM T02565 D0C4RB 36314 IC50 = 260 nM T02565 D0G3DL 135398735 Ki = 1400 nM T02565 D0MY8N 5280489 Ki = 2260 nM T02565 D0N6RF 65999 Ki = 960 nM T02565 D0R1RS 3715 Ki = 38000 nM T02565 D0R3JB 4212 Ki = 3100 nM T02565 D0V8QT 2708 Ki = 37400 nM T02565 D0W9MM 13342 Ki = 18600 nM T02565 D0Z1ZM 84029 IC50 = 3311.31 nM T02565 D0ZU9R 392622 Ki = 4000 nM T02565 D0C5VQ 1548994 IC50 = 5000 nM T02565 D0CE0O 11513676 IC50 = 220 nM T02565 D0G7UX 5284373 Ki = 1200 nM T02565 D0L4FS 5280961 Ki = 2960 nM T02565 D0V1WQ 24857286 IC50 = 11200 nM T02565 D0Z0HH 3503 Ki = 3470 nM T02565 D0G6ZW 636402 Ki = 1480 nM T02565 C5Q6US 2540 Ki = 1900 nM T02565 CT6YF0 5100 Ki = 3150 nM T02565 C2AMP7 25096 Ki = 940 nM T02565 CYQ4S7 60822 Ki = 2580 nM T02565 CXJV17 73157 Ki = 1250 nM T02565 CQD56Z 73299 Ki = 680 nM T02565 C4HU6M 92095 Ki = 80 nM T02565 CNIW58 107905 Ki = 3460 nM T02565 CW90BT 441336 Ki = 870 nM T02565 C82BDA 441371 Ki = 2350 nM T02565 CI4K8B 443953 Ki = 1610 nM T02565 CT2W6J 467315 Ki = 6500 nM T02565 C76DRY 638034 Ki = 3890 nM T02565 CAW27Q 3503223 Ki = 1840 nM T02565 C8B3NE 4565183 Ki = 2020 nM T02565 CT5ZR8 5149276 Ki = 1770 nM T02565 CNI9X4 5281888 Ki = 5900 nM T02565 CM47KI 5351344 IC50 = 194540 nM T02565 CH9WV2 5379540 Ki = 420 nM T02565 C46NFC 6426773 Ki = 590 nM T02565 CGVZ63 6708545 Ki = 600 nM T02565 C81NYO 6857763 Ki = 560 nM T02565 CAV9Q8 6857785 Ki = 3940 nM T02565 CPIV47 6857789 Ki = 4170 nM T02565 C6ROL5 6857793 Ki = 2240 nM T02565 CF5M6V 6857794 Ki = 1730 nM T02565 CI28JY 10457775 IC50 > 200000 nM T02565 CSH8G0 10960835 Ki = 2890 nM T02565 C7TKI8 21596329 Ki = 3060 nM T02565 CM5P2W 21633776 Ki = 2920 nM T02565 CYK84S 23675786 Ki = 1550 nM T02565 CHJP54 23681233 Ki = 2710 nM T02565 C9P5GD 23703990 Ki = 3310 nM T02565 CPM3X9 24721251 Ki = 4020 nM T02565 CZ8SR1 40469657 Ki = 5990 nM T02565 CTE19R 40469671 IC50 = 3235.94 nM T02565 CKI50V 40469815 Ki = 3810 nM T02565 C70JTD 44575959 Ki = 2610 nM T02565 CU49XY 52947716 Ki = 440 nM T02565 CM09JD 54676535 Ki = 560 nM T02565 CPE5F1 73348206 Ki = 2670 nM T02565 CLAF78 73354262 Ki = 6590 nM T02565 CRT3Q7 76311369 Ki = 2160 nM T02565 C19WRY 76311434 Ki = 3050 nM T02565 CU76LZ 76313482 Ki = 2630 nM T02565 CBLK75 76315020 Ki = 1080 nM T02565 C7XM6W 76322315 IC50 = 2951.21 nM T02565 CZ8AR0 76322316 Ki = 2270 nM T02565 C7W1VB 76325939 Ki = 2390 nM T02565 CR6QG3 76333163 Ki = 3470 nM T02565 C0T3XF 76333164 Ki = 2550 nM T02565 CE61WT 76333166 Ki = 2890 nM T02565 CQ9E0I 76336791 Ki = 2890 nM T02565 COVK20 90142631 IC50 = 880 nM T02565 CFB4D9 135403795 Ki = 3420 nM T02565 C7GK3H 145990715 IC50 = 39490 nM T02565 D04LBT 14957 Ki = 3820 nM T02565 D07LUJ 64945 IC50 = 11481.54 nM T02565 D0F2AD 119245 Ki = 1030 nM T02565 D0G2JZ 1464 Ki = 16000 nM T02565 D0HD9P 444899 Ki = 820 nM T02565 D0J5RQ 234102 IC50 = 11481.54 nM T02565 D0O8ZV 5280352 Ki = 2630 nM T02565 D0R4WJ 16129778 Ki = 3230 nM T02565 D0U8IF 10114 Ki = 420 nM T02565 D0UQ6U 10569 Ki = 4080 nM T79780 D0V2GT 5311023 Ki = 12 nM T79780 C2H5NY 9854861 EC50 = 158.49 nM T79780 C3H7AS 9955930 Ki = 23 nM T79780 CH1Q6E 10008757 Ki = 1100 nM T79780 C6S2CB 25138123 IC50 = 640 nM T79780 CMTA17 44542176 EC50 = 527 nM T79780 COW17D 44542178 EC50 = 2370 nM T79780 C7Q9PI 44542320 EC50 = 794.33 nM T79780 C3ILH8 44542324 EC50 = 79.43 nM T79780 C8D4AT 44542326 EC50 = 158.49 nM T79780 CIRQ85 44542328 EC50 = 39.81 nM T79780 CB58DA 44542330 EC50 = 125.89 nM T79780 CS12HR 44542332 EC50 = 316.23 nM T79780 CY4L2G 53318788 IC50 = 1.9 nM T79780 CO72VY 60168134 EC50 = 4608 nM T79780 CH58GJ 71450762 Ki = 15 nM T79780 C6AV0I 71451611 EC50 = 1.7 nM T79780 C7K8BZ 71452593 Ki = 35 nM T79780 COM10Q 71454352 Ki = 29 nM T79780 CM31QR 71454353 Ki = 114 nM T79780 CL9E0V 71454357 Ki = 110 nM T79780 C8MP1A 71454358 Ki = 2 nM T79780 CHFO89 71454359 Ki = 167 nM T79780 C7ROU1 71456101 Ki = 0.8 nM T79780 CO07CE 71456102 Ki = 84 nM T79780 C24UFT 71456103 Ki = 121 nM T79780 CL82IR 71456104 Ki = 6 nM T79780 C3SOE7 71457908 Ki = 378 nM T79780 CZ7C4L 71457909 Ki = 10 nM T79780 CJWQ68 71457910 Ki = 5 nM T79780 C3W7BS 71461185 Ki = 198 nM T79780 C0VA5C 71463271 Ki = 87 nM T79780 C5GN8U 71463272 Ki = 0.9 nM T79780 C49KZP 71463273 Ki = 51 nM T79780 C1EGB8 71463275 Ki = 273 nM T79780 CW9XZ8 71463276 Ki = 106 nM T79780 CA7S8C 71463277 Ki = 0.32 nM T79780 C75FXY 71463278 Ki = 2 nM T79780 CA7G4S 71463279 Ki = 11 nM T79780 C4VM7N 90324505 EC50 > 5000 nM T79780 C2AY1B 90324535 EC50 > 5000 nM T79780 CW3LH2 101882818 Ki = 487 nM T79780 CW5H9D 101882819 Ki = 81 nM T79780 CGQV37 101882820 Ki = 112 nM T79780 CA51CQ 118724536 Ki = 58 nM T79780 CR4MG1 118724537 Ki = 3.85 nM T79780 CBA2Z0 118724538 Ki > 5000 nM T79780 CL3T4A 118724539 Ki = 2906 nM T79780 CTHD48 118724540 Ki = 479 nM T79780 CZL32K 118724541 Ki > 5000 nM T79780 C5HNX2 118724542 Ki = 1880 nM T79780 C4AT2F 118724543 Ki = 2965 nM T79780 CE1NT2 118724544 Ki > 5000 nM T79780 CM3RN4 118724970 Ki = 441 nM T79780 C5XD1N 118724971 Ki = 3429 nM T79780 C6M1AZ 118724972 Ki = 2692 nM T79780 CSF21L 118724973 Ki = 2454 nM T79780 CH4LB0 118724977 Ki = 319 nM T79780 C6GK5N 118724978 Ki = 904 nM T79780 C9SN0M 118724979 Ki = 94 nM T79780 CH9GT5 118724980 Ki = 114 nM T79780 CHK0S7 118724981 Ki = 201 nM T79780 C1BVC2 118724982 Ki = 191 nM T79780 C76XZK 118724983 Ki = 511 nM T79780 CG7SQ8 118724984 Ki = 417 nM T79780 CB3D6X 118724985 Ki = 151 nM T79780 CG04KW 118724986 Ki = 15085 nM T79780 CO69YD 118724987 Ki = 1638 nM T79780 C72AKO 118724988 Ki = 1057 nM T79780 C4CRS0 118724989 Ki = 538 nM T79780 CJIB02 118724990 Ki = 141 nM T79780 CD41AL 118724991 Ki = 112 nM T79780 C2DCZ3 118724992 Ki = 340 nM T79780 C49HSM 118724993 Ki = 432 nM T79780 CE9ZS5 118724994 Ki = 316 nM T79780 CP2WY4 118724995 Ki = 296 nM T79780 CE1LW7 118735685 EC50 = 222 nM T79780 C5PA2G 127041908 Ki = 630 nM T79780 C62JIE 127042244 Ki = 1000 nM T79780 CNX9D2 136948074 Ki = 1966 nM T79780 CY35MT 136998789 Ki = 1623 nM T79780 CBAP98 136998790 Ki = 2348 nM T79780 C8F9WQ 155515973 IC50 = 190 nM T79780 CF42WX 155520785 IC50 = 520 nM T79780 D01VSI 25240297 IC50 = 4.7 nM T79780 D08UWO 53320361 Ki = 22 nM T79780 D0JE3Z 16735569 IC50 = 160 nM T02392 D05UFG 10184653 IC50 > 10000 nM T02392 D0O8GK 71496458 IC50 = 32900 nM T02392 D0J6AU 10152654 IC50 > 10 nM T02392 D0YB3W 156414 IC50 = 2700 nM T02392 D0HM5J 118253852 IC50 = 3.981 nM T02392 C0XQP7 6917747 IC50 > 100000 nM T02392 CD54AH 6993099 Ki = 6200000 nM T02392 CBS6P7 8022437 IC50 = 11000 nM T02392 CXE30M 11334066 IC50 = 822 nM T02392 C9D6XI 11736400 IC50 = 172 nM T02392 C8D7BS 11771234 IC50 = 13 nM T02392 CN4IM8 11817961 IC50 = 96 nM T02392 C31MCN 13186896 IC50 > 100000 nM T02392 C6XPN4 16664855 IC50 = 18 nM T02392 CZ8DI1 23643986 IC50 = 70 nM T02392 CZPF48 23648277 IC50 > 10000 nM T02392 C31XJH 23648296 IC50 > 10000 nM T02392 CN0VA7 24822701 IC50 = 14 nM T02392 CQU38W 24900755 IC50 = 1727 nM T02392 C2S8VB 24901099 IC50 = 29 nM T02392 CIN28B 24901100 IC50 = 403 nM T02392 CD2EH0 24901101 IC50 = 191 nM T02392 CS7B3F 24901102 IC50 > 10000 nM T02392 CGI0U2 25023791 Ki = 10000 nM T02392 C3C8YJ 25174148 IC50 = 1.995 nM T02392 C5M1BT 25195691 IC50 = 158.49 nM T02392 CJ63ZU 42641779 IC50 = 158.49 nM T02392 CZM36T 42641892 IC50 = 39.81 nM T02392 CRYH80 42642459 IC50 = 1 nM T02392 C25ELB 44143088 IC50 = 34.67 nM T02392 CL0M7R 44143089 IC50 = 6918.31 nM T02392 C9QDC0 44143091 IC50 = 588.84 nM T02392 CDVC01 44268431 Ki = 180000 nM T02392 CK8EB3 44268436 Ki = 220000 nM T02392 CAPM01 44413250 IC50 = 6296 nM T02392 C7EKG5 44413251 IC50 = 9637 nM T02392 CCG5S4 44413390 IC50 = 137 nM T02392 CS6X7V 44426055 IC50 = 606 nM T02392 C8IB2W 44426056 IC50 > 100000 nM T02392 C9TFJ8 44464926 IC50 = 10 nM T02392 CYO0T1 44465454 IC50 = 7.943 nM T02392 CE83YL 44465721 IC50 < 0.3981 nM T02392 C6OC4Z 44607530 IC50 = 2100 nM T02392 CWMN69 46882864 IC50 = 2545 nM T02392 CQT8N7 46882865 IC50 = 271 nM T02392 CP47RN 46882866 IC50 = 8.2 nM T02392 C75BEM 46882867 IC50 = 1.7 nM T02392 C2PKZ9 46882868 IC50 = 880 nM T02392 CLV43E 46882869 IC50 = 336 nM T02392 CY2MQ1 46882870 IC50 = 2193 nM T02392 C0M4PL 46882914 IC50 = 250 nM T02392 CC94XY 46882915 IC50 = 67 nM T02392 C5X4SE 46883366 IC50 = 1230 nM T02392 CO5PD8 46883367 IC50 = 29 nM T02392 C9J4KG 46883368 IC50 = 5.8 nM T02392 CNA0W6 46883391 IC50 = 200 nM T02392 CW1RB0 46883392 IC50 = 630 nM T02392 CEB8W0 46883393 IC50 = 1580 nM T02392 CXST57 46883394 IC50 = 330 nM T02392 C7I6OU 46883395 IC50 = 17 nM T02392 CA6BD2 46883396 IC50 = 215 nM T02392 CP0V2B 46883425 IC50 = 3.8 nM T02392 C4WNV1 46883426 IC50 = 5.1 nM T02392 C16KZC 46883427 IC50 = 0.9 nM T02392 CQX57K 46883428 IC50 = 11 nM T02392 CQN34G 46883429 IC50 = 1 nM T02392 C0ZH2Y 46883430 IC50 = 0.7 nM T02392 C56QYZ 46883464 IC50 = 0.3 nM T02392 CEZ54V 46883465 IC50 > 3000 nM T02392 C2QM7R 46883466 IC50 = 12 nM T02392 CE80HK 46883467 IC50 = 1419 nM T02392 CHA61U 46883468 IC50 = 1832 nM T02392 CI2FX9 46883469 IC50 = 63 nM T02392 CM4O6Q 46883470 IC50 = 17 nM T02392 C68XTP 46883502 IC50 = 2502 nM T02392 CYN9C1 46883503 IC50 = 1081 nM T02392 C6FI5J 46883504 IC50 = 495 nM T02392 C7IOX5 46883505 IC50 = 133 nM T02392 C3I0FZ 46883506 IC50 > 10000 nM T02392 CUI91D 46905615 IC50 > 220 nM T02392 C9PAR7 46905616 IC50 = 790 nM T02392 CAFW31 49783666 IC50 = 0.7943 nM T02392 CN0B1V 49783830 IC50 = 0.2512 nM T02392 CNI1P6 49783903 IC50 = 0.7943 nM T02392 CGF65B 49783985 IC50 = 5.012 nM T02392 CI59MV 49797572 IC50 > 30000 nM T02392 C96CKU 49797573 IC50 = 14 nM T02392 C56OCA 53317528 IC50 = 1995.26 nM T02392 C7I9AO 53317529 IC50 > 25118.86 nM T02392 CM60RJ 53317530 IC50 > 25118.86 nM T02392 C5A6IH 53317737 IC50 = 1000 nM T02392 C6FEH9 53318816 IC50 > 25118.86 nM T02392 CJAX07 53318817 IC50 = 15848.93 nM T02392 CG5AP6 53318818 IC50 = 125.89 nM T02392 C0QV5D 53322753 IC50 = 2511.89 nM T02392 CHB96K 53324300 IC50 = 316.23 nM T02392 CR1L4Y 53325394 IC50 > 25118.86 nM T02392 CVU0J1 53326656 IC50 = 316.23 nM T02392 CFC91M 54769914 IC50 = 2.512 nM T02392 CF3XA9 57999656 IC50 = 158.49 nM T02392 CLA3R9 66645269 IC50 = 1.995 nM T02392 C62SML 90655967 IC50 = 25.12 nM T02392 CJ7LT3 90655968 IC50 = 12.59 nM T02392 CB61WC 90655969 IC50 = 3.981 nM T02392 CK5X2M 91826235 IC50 = 2.512 nM T02392 CGFK60 101201806 IC50 = 51 nM T02392 C8E4WS 102323332 IC50 = 1 nM T02392 CI9L7M 118253811 IC50 = 15.85 nM T02392 C3BAX2 118253818 IC50 = 6309.57 nM T02392 CL5C4K 118253824 IC50 = 7.943 nM T02392 CO53KU 118253851 IC50 = 12.59 nM T02392 C7YFQ0 118253855 IC50 = 15.85 nM T02392 CCH97D 118253857 IC50 = 31.62 nM T02392 C24IWU 118253859 IC50 = 39.81 nM T02392 CM63RL 118253870 IC50 = 12.59 nM T02392 CPBD92 118253877 IC50 = 63.1 nM T02392 CCG7Y6 118253883 IC50 = 5.012 nM T02392 CA72QZ 118253888 IC50 = 6.31 nM T02392 C63BSU 118260121 IC50 = 63.1 nM T02392 CTE34I 118720232 IC50 > 100000 nM T02392 CSD62B 118720233 IC50 > 100000 nM T02392 C9WF7Q 118720234 IC50 = 66000 nM T02392 C76HIO 118720235 IC50 = 18000 nM T02392 CAT1R6 118720236 IC50 > 100000 nM T02392 CGAF42 118720237 IC50 > 100000 nM T02392 CJ28KZ 118720238 IC50 > 100000 nM T02392 CPH2V9 118720239 IC50 > 100000 nM T02392 CQA83T 134131850 IC50 = 199.53 nM T02392 C7UNJ4 134132070 IC50 > 10000 nM T02392 CVAH73 134134180 IC50 = 398.11 nM T02392 CD6H8U 134134303 IC50 > 10000 nM T02392 C1RWN0 134134473 IC50 = 1000 nM T02392 CB93JM 134134976 IC50 = 1258.93 nM T02392 CZL0G9 134138927 IC50 = 158.49 nM T02392 C1W7EY 134140481 IC50 = 501.19 nM T02392 C6B5RW 134141023 IC50 = 39.81 nM T02392 CO9E0J 134145021 IC50 = 25.12 nM T02392 CI6FZ3 134147640 IC50 > 10000 nM T02392 C3DCQ9 134148503 IC50 = 501.19 nM T02392 C9OLA1 134148630 IC50 > 10000 nM T02392 C8SH1L 134154191 IC50 = 31.62 nM T02392 CTQY96 136117851 IC50 = 450 nM T02392 C3YHN7 146685679 IC50 = 32.3 nM T02392 C7TI5V 147202641 IC50 > 10000 nM T02392 CIK2C0 147243243 IC50 = 2150 nM T02392 C0JL2F 147323358 IC50 = 4 nM T02392 CUAY08 148018738 IC50 = 12.3 nM T02392 CH0NR2 148192765 IC50 > 10000 nM T02392 CT25HK 148412521 IC50 = 2.7 nM T02392 CWD7A1 148809433 IC50 = 2051 nM T02392 C0SW6H 148967294 IC50 = 6.5 nM T02392 CQK39B 149491764 IC50 = 3.9 nM T02392 C1ZX5D 149494192 IC50 = 1.9 nM T02392 CCU10W 149589615 IC50 = 505 nM T02392 CN6G2P 149839762 IC50 = 307.1 nM T02392 C4GCQ2 149933110 IC50 > 10000 nM T02392 C08LSG 150088178 IC50 = 154 nM T02392 CJZ3L2 150363449 IC50 = 783 nM T02392 C26MXO 150396261 IC50 = 1520 nM T02392 C3IPK7 150631495 IC50 = 271 nM T02392 CJ6A9B 150967523 IC50 = 221 nM T02392 CFXO59 151118910 IC50 = 499 nM T02392 CO6QT1 151217326 IC50 = 2.8 nM T02392 CMX4K7 151268438 IC50 = 4.9 nM T02392 CG6CN4 151286177 IC50 = 1605 nM T02392 C7RZO2 151821865 IC50 = 785 nM T02392 CDL4W5 151971947 IC50 = 1 nM T02392 CYN8L2 152157601 IC50 = 537 nM T02392 CJ2KV5 152225461 IC50 = 135.4 nM T02392 CKZ6H9 152242423 IC50 = 21.3 nM T02392 COE18M 152296790 IC50 = 175 nM T02392 CR0EQ1 152335936 IC50 = 835 nM T02392 C0IO7L 152457310 IC50 = 391.5 nM T02392 CZG2D5 152823047 IC50 = 2.3 nM T02392 CPF6I5 155518852 IC50 = 483 nM T02392 CQF3W2 155521718 IC50 > 10000 nM T02392 CXC8Q2 155522247 IC50 = 79.43 nM T02392 CMJO87 155528739 IC50 = 630.96 nM T02392 CY2HC7 155538869 IC50 = 6.31 nM T02392 CVGT48 155543410 IC50 = 0.3981 nM T02392 C2J5NY 155559747 IC50 = 50.12 nM T02392 CU67FS 155561515 IC50 = 50.12 nM T02392 CA8WQ7 155565392 IC50 = 1.585 nM T02392 D00FGA 73737 IC50 > 25118.86 nM T02392 D09FGQ 123985 IC50 = 770 nM T02392 D0IV5D 11241135 Ki = 2700 nM T02392 D0L9VP 5287864 IC50 = 2600 nM T02392 D0U4TA 44413276 IC50 = 4787 nM T02392 D0Y5IQ 44255320 IC50 = 10000 nM T93266 D06TKE 9796088 IC50 = 158.49 nM T93266 CV27NR 16015404 IC50 = 398.11 nM T93266 CC2UO9 16015637 IC50 > 199526.23 nM T93266 CQ62LZ 16803385 IC50 = 2511.89 nM T93266 CY59DU 17616875 IC50 > 199526.23 nM T93266 CD3A1C 35579115 IC50 = 31.62 nM T93266 CV84AF 39734391 IC50 > 199526.23 nM T93266 CC50GL 39734394 IC50 = 125.89 nM T93266 CU98ZN 53386723 IC50 = 398.11 nM T93266 CDG90A 56658576 IC50 = 15.85 nM T93266 CK9BH7 56658685 IC50 = 50118.72 nM T93266 C40VQA 56662019 IC50 = 15848.93 nM T93266 CY76ZF 56662020 IC50 = 398.11 nM T93266 C06MAF 56662154 IC50 = 1258.93 nM T93266 C36LWN 56662155 IC50 = 630.96 nM T93266 CC67MA 56662156 IC50 = 25118.86 nM T93266 C91VWQ 56662157 IC50 = 630.96 nM T93266 C41JXW 56665509 IC50 = 316.23 nM T93266 C48YMD 56665613 IC50 = 25118.86 nM T93266 C5GPD3 56665614 IC50 = 63095.73 nM T93266 CLH3F2 56668937 IC50 = 50.12 nM T93266 CC41RK 56668938 IC50 = 79.43 nM T93266 CE87DY 56672420 IC50 = 31.62 nM T93266 CU8TA0 56672421 IC50 > 199526.23 nM T93266 CZMJ98 56672531 IC50 = 398.11 nM T93266 CEBM89 56672532 IC50 = 63095.73 nM T93266 CE0LI2 56672533 IC50 = 19952.62 nM T93266 CBVO32 56675803 IC50 = 251.19 nM T93266 C91FGR 56675804 IC50 = 199.53 nM T93266 CX5I9D 56675805 IC50 = 1584.89 nM T93266 C6GLB7 56675914 IC50 > 199526.23 nM T93266 CW4S7Z 56679123 IC50 = 630.96 nM T93266 CE4H6B 56679227 IC50 = 100000 nM T93266 C7WCZ1 56679228 IC50 = 15848.93 nM T93266 C68OFP 56682419 IC50 > 199526.23 nM T47164 D0OB0F 5328940 IC50 = 191 nM T47164 D0E3TC 44259 IC50 = 1.58 nM T47164 D03BNU 59604787 IC50 > 10000 nM T47164 D0T3ME 156422 IC50 > 30000 nM T47164 CACS26 11561968 Ki > 2000 nM T47164 CU0E8O 11690457 Ki > 2000 nM T47164 CC71QJ 27666048 IC50 > 100000 nM T47164 C3VRO9 44557921 IC50 > 10000 nM T47164 C8NA4L 53384644 IC50 > 30000 nM T47164 C1MR8Q 60097495 IC50 > 1000 nM T47164 CV63UL 67240318 IC50 > 10000 nM T47164 C2AN7T 134611886 IC50 > 100000 nM T47164 C6VB3O 145925651 IC50 >= 5000 nM T47164 C8V1GD 154853229 IC50 > 10000 nM T47164 C2MD1Q 155513187 IC50 > 10000 nM T35565 D0G7IY 27503 IC50 = 9680000 nM T35565 D00YPW 135399235 IC50 = 6250000 nM T35565 C57OTC 13818 Ki = 11000000 nM T35565 C7H9AN 52780 IC50 = 1200 nM T35565 C7GTI4 81312 Ki = 580000 nM T35565 C6OY2Q 173894 IC50 = 100000 nM T35565 CDV2A5 197063 Ki = 19000000 nM T35565 CD3JC2 198439 IC50 = 350000 nM T35565 CA0ZS6 204484 Ki = 1550000 nM T35565 CTQ78Z 646625 IC50 = 800000 nM T35565 CA09QJ 715454 IC50 = 600 nM T35565 CI4B6F 3047246 IC50 = 160000 nM T35565 C5GWL4 3047254 IC50 = 180000 nM T35565 CK41ZQ 10379025 Ki = 1500000 nM T35565 C0C5MW 10877388 Ki = 40000 nM T35565 CSN84C 10880008 Ki = 390000 nM T35565 CNR8J4 10921447 Ki = 7000000 nM T35565 C1SO8X 11031366 Ki = 460000 nM T35565 C80KUM 11151757 Ki = 330000 nM T35565 CYB81K 11183084 Ki = 200000 nM T35565 C1D4YC 12124355 Ki = 1500000 nM T35565 CBFR34 12473031 IC50 = 170000 nM T35565 CXRP20 12473033 IC50 = 710000 nM T35565 C9CH7I 12512356 IC50 = 280000 nM T35565 CN9B2D 12512360 IC50 = 410000 nM T35565 C5ROA6 12512364 IC50 = 220000 nM T35565 C6OU2Y 12762400 IC50 = 620000 nM T35565 C56OQB 12762401 IC50 = 230000 nM T35565 C42ISG 13019718 IC50 = 140000 nM T35565 CJ50DX 13019728 IC50 = 280000 nM T35565 CG75IB 13019729 IC50 = 210000 nM T35565 CD67HQ 13019730 IC50 = 340000 nM T35565 C23AXE 13019731 IC50 = 230000 nM T35565 CEI89B 20262261 Ki = 600000 nM T35565 CQU54I 20555046 IC50 > 10000000 nM T35565 C7RI9A 25067484 IC50 = 1700 nM T35565 CM1SX9 25067486 IC50 = 6200 nM T35565 CDJX98 25067492 IC50 = 30500 nM T35565 CG3LC6 25067494 IC50 = 2700 nM T35565 CN67WC 25067496 IC50 = 9400 nM T35565 C8G0HM 44377473 IC50 > 10000000 nM T35565 D0RC4F 72103 IC50 = 970000 nM T21661 C2UX5G 25270307 IC50 = 87910 nM T21661 C79IOK 25270309 IC50 = 27830 nM T21661 C59TRU 25270648 IC50 = 21000 nM T21661 CHO82Q 25270650 IC50 = 1430 nM T21661 CL3S5V 25270986 IC50 = 15870 nM T21661 C7KSO5 71449539 IC50 > 100000 nM T21661 CJ6SQ8 71451328 IC50 > 100000 nM T21661 C2F5XK 71453144 IC50 = 66380 nM T21661 CTP47E 71454881 IC50 = 55000 nM T21661 CB1WD6 71456658 IC50 = 8110 nM T21661 CSU17Q 71460350 IC50 > 100000 nM T21661 C0UXW2 71462049 IC50 > 100000 nM T21661 C7FEJ4 71462050 IC50 = 1730 nM T63159 D0RA5Q 72172 Ki = 190 nM T63159 CYQ8J7 9849506 IC50 = 854 nM T63159 CTZQ69 10347030 IC50 = 2503 nM T63159 CAIN04 10851204 IC50 = 790 nM T63159 CVZ7S9 12945733 Ki = 43 nM T63159 C59KCI 16066739 IC50 = 1149 nM T63159 CD85RP 16114636 IC50 = 91 nM T63159 CWS8E9 16114761 IC50 = 406 nM T63159 CEK6O8 16114767 IC50 = 45 nM T63159 CC5G9I 16114887 IC50 = 41 nM T63159 CN0KE7 16114891 IC50 = 1931 nM T63159 CC2TL6 16115011 IC50 = 107 nM T63159 CM29PA 16115017 IC50 = 253 nM T63159 CF59ML 16115018 IC50 = 1760 nM T63159 C7UD5V 16115131 IC50 = 206 nM T63159 C4Q5ZG 16115133 IC50 = 5363 nM T63159 CS20KE 16115134 IC50 = 1168 nM T63159 C3A6BL 16115135 IC50 = 2515 nM T63159 CMP8B2 16115136 IC50 = 164 nM T63159 CKA40L 16115137 IC50 = 130 nM T63159 C98HRF 16115247 IC50 = 231 nM T63159 CJ89VD 16115252 IC50 = 527 nM T63159 C83IPC 16115366 IC50 = 225 nM T63159 CASZ30 16115370 IC50 = 966 nM T63159 CA4NX9 16115494 IC50 = 248 nM T63159 CQ0V6G 16115921 IC50 = 6 nM T63159 CO6S2Z 16115922 IC50 = 13 nM T63159 C9O1WK 16115923 IC50 = 330 nM T63159 C5O6LK 16116059 IC50 > 10000 nM T63159 C31AOC 16116060 IC50 > 10000 nM T63159 CP9TA2 16116577 IC50 = 904 nM T63159 CLX59A 16116578 IC50 = 3896 nM T63159 CJ8L6N 44323514 IC50 > 10000 nM T63159 C7K8JV 44323547 IC50 = 1540 nM T63159 CRAI45 44323558 IC50 = 21000 nM T63159 C5H4PG 44420648 IC50 = 109 nM T63159 CHC38Q 50919282 Ki = 490 nM T63159 CH1F8E 51355980 Ki = 900 nM T63159 C6ZX3T 51356259 Ki = 1450 nM T63159 CDT9C4 51356260 Ki > 15000 nM T63159 CWN17C 51356261 Ki > 15000 nM T63159 CPK49Y 51356262 Ki > 15000 nM T63159 C7KXV5 51356561 Ki = 3000 nM T63159 C6DHM3 51356564 Ki = 5300 nM T63159 C7SV3D 101874839 Ki = 0.7 nM T63159 C9W6XA 101874840 Ki = 5.5 nM T63159 CZ0CF5 101874841 Ki = 7.4 nM T63159 CE03QN 118723770 Ki > 500 nM T63159 C8KZV5 118723771 Ki > 500 nM T63159 C95ZHI 118723772 Ki = 0.8 nM T63159 CMWK83 118723773 Ki = 74.5 nM T63159 C2R0AF 118723775 Ki = 113 nM T63159 CX9PR0 118723776 Ki = 41.3 nM T63159 CUWD14 118723777 Ki = 12.3 nM T63159 C16MZO 118723778 Ki = 15.3 nM T63159 C5A4ZW 118723779 Ki = 23 nM T63159 CH4AJ6 118723780 Ki = 1.9 nM T63159 C14NYA 118723781 Ki = 4 nM T63159 CNO5J0 118723782 Ki = 11.2 nM T63159 D01LFP 16114883 IC50 = 170 nM T63159 D06TVS 16116576 IC50 = 495 nM T63159 D0D8FZ 16114889 IC50 = 1011 nM T63159 D0GB8I 16114635 IC50 = 885 nM T63159 D0K9XV 16114884 IC50 = 57 nM T63159 D0YA8C 10592233 IC50 = 125 nM T63159 D0YO0R 16115012 IC50 = 46 nM T63159 D0Z2JN 10709191 IC50 = 125 nM T10147 D0I2AN 86298439 IC50 = 8600 nM T10147 CW68ZS 61672 IC50 = 10000 nM T10147 CGF5Q9 5281701 IC50 = 17500 nM T10147 C53RWT 5393164 IC50 = 3000 nM T10147 CM8I0N 5781144 IC50 = 500 nM T10147 CJG32W 56659993 IC50 = 5200 nM T10147 C2WDB7 56680468 IC50 = 3600 nM T10147 C2MX8E 56683798 IC50 = 4300 nM T10147 C7LQ6J 57405802 IC50 = 6600 nM T10147 CW2FZ3 68075819 IC50 = 4600 nM T10147 CSL3N8 68075861 IC50 = 6300 nM T10147 CPY5S8 68075863 IC50 = 6100 nM T10147 C6KR0D 122194839 IC50 = 15600 nM T10147 C85FQM 122194840 IC50 = 11800 nM T10147 C6SIU3 122194841 IC50 = 7900 nM T10147 CX2Y3K 122195056 IC50 = 600 nM T10147 CR6P8H 122195057 IC50 = 900 nM T10147 C4IUQ6 127040400 IC50 = 800 nM T10147 CB5S6H 127041739 IC50 = 900 nM T10147 C1DEH7 127042038 IC50 = 5400 nM T10147 CTY0E4 127042039 IC50 = 10400 nM T10147 C8BG3P 155564911 IC50 = 38000 nM T10147 D00LMG 5281697 IC50 = 600 nM T10147 D00YEV 5281605 IC50 = 10300 nM T10147 D0NJ4H 5281670 IC50 = 4300 nM T01255 D0E3TC 44259 IC50 = 49.1 nM T01255 CV63UL 67240318 IC50 > 10000 nM T01255 C2MD1Q 155513187 IC50 > 10000 nM T63505 D00STL 644241 IC50 < 2.54 nM T63505 D01PZD 5329098 IC50 = 11000 nM T63505 D01ZRI 6450551 IC50 = 1 nM T63505 D03MNN 11341869 IC50 = 0.4 nM T63505 D03ZBT 11626560 IC50 = 1159 nM T63505 D04LVK 57379345 IC50 = 1250 nM T63505 D07POC 176870 IC50 = 2100 nM T63505 D07TOK 46188928 IC50 > 1000 nM T63505 D08CDI 208908 IC50 = 23000 nM T63505 D09XZB 123631 IC50 = 1200 nM T63505 D0AZ3C 5291 Ki = 13 nM T63505 D0C4RB 36314 IC50 > 10000 nM T63505 D0E6XR 3062316 Ki = 0.457 nM T63505 D0E7PQ 5311 IC50 > 100000 nM T63505 D0G6QF 3081361 IC50 = 86 nM T63505 D0H0EQ 24826799 IC50 = 0.32 nM T63505 D0J1MI 4030 Ki = 4600 nM T63505 D0J9ZR 4477 IC50 > 100000 nM T63505 D0OB0F 5328940 IC50 = 1.1 nM T63505 D0R0MW 5329102 IC50 = 410 nM T63505 D0W5HK 216239 IC50 = 120 nM T63505 D00DRL 44137946 IC50 = 7800 nM T63505 D00UZR 5330286 IC50 > 10000 nM T63505 D02RJY 11442891 IC50 = 5 nM T63505 D02XNW 5494449 Ki = 30 nM T63505 D03HUX 49792852 IC50 > 10000 nM T63505 D03LWG 53235510 IC50 = 2300 nM T63505 D04AHQ 71721540 IC50 = 380 nM T63505 D05ADP 160355 IC50 > 10000 nM T63505 D05PZB 135398495 IC50 = 4 nM T63505 D06DMQ 59472121 Ki = 59 nM T63505 D07DTV 11338033 IC50 > 10000 nM T63505 D07EHV 44814409 IC50 > 10000 nM T63505 D07HPJ 11476171 IC50 > 10000 nM T63505 D08HOM 46207586 IC50 = 12 nM T63505 D0CY1B 6420138 Ki > 10000 nM T63505 D0E3TC 44259 IC50 = 30 nM T63505 D0G0VV 11387605 IC50 = 26 nM T63505 D0L4FS 5280961 IC50 = 10000 nM T63505 D0M0XB 10302451 IC50 = 30 nM T63505 D0O0LS 25141092 IC50 > 1000 nM T63505 D0P1CV 46191454 IC50 > 10000 nM T63505 D0Q9UX 16718576 IC50 = 478 nM T63505 D0S7HM 16041424 IC50 = 81 nM T63505 D0Z4RC 24756910 IC50 = 2890 nM T63505 D03BNU 59604787 IC50 > 10000 nM T63505 D01KIJ 72545600 IC50 = 0.7 nM T63505 D01LMW 89899422 IC50 = 166 nM T63505 D0EF5T 44129660 IC50 = 17 nM T63505 D0JY1I 42613483 IC50 = 1800 nM T63505 D0OE4F 4369496 IC50 = 100 nM T63505 D0Y9PK 53346432 Ki > 15000 nM T63505 D01EFO 9864718 IC50 = 400 nM T63505 D0Q7HO 4705 IC50 = 30 nM T63505 D0T3ME 156422 IC50 = 41000 nM T63505 CB1VW3 1400 IC50 = 147 nM T63505 C8KF1N 4122 IC50 = 640 nM T63505 CJ17AM 4877 IC50 = 7 nM T63505 CBPM40 4878 Ki = 500 nM T63505 CFA4M1 40320 Ki = 10000 nM T63505 C6SB2N 123596 IC50 = 430 nM T63505 C6Y9CV 151193 IC50 > 10000 nM T63505 C9WA8F 341040 IC50 > 100000 nM T63505 C3MS0Y 346935 IC50 = 10000 nM T63505 CC2R6G 409975 IC50 > 100000 nM T63505 CB9F1O 447961 Ki = 160 nM T63505 C13HGZ 644784 Ki = 360 nM T63505 C02LNV 644846 Ki = 90 nM T63505 CP1H6K 660311 IC50 = 251.19 nM T63505 CLV7T4 685639 Ki = 70 nM T63505 C0TK5Y 726259 Ki = 624 nM T63505 CBQ69T 741735 IC50 = 158.49 nM T63505 C7P9XJ 779445 Ki = 16 nM T63505 C4PU1I 809029 Ki = 278 nM T63505 C39HTG 825387 Ki = 58000 nM T63505 C2YQW4 854410 IC50 = 12589.25 nM T63505 C63EYU 889490 Ki = 68 nM T63505 CA2X3D 1049031 Ki = 20000 nM T63505 C8AOR6 1113641 Ki = 97 nM T63505 CX78TH 1113642 Ki = 249 nM T63505 CD3IH5 1143580 Ki = 136 nM T63505 CTL80W 1312422 IC50 = 251.19 nM T63505 CQR4S9 1327207 Ki = 47 nM T63505 CQ47RP 1358652 IC50 = 398.11 nM T63505 C1RQ4E 1886699 IC50 = 74000 nM T63505 C6NK9W 1898760 IC50 = 72000 nM T63505 CRZ40I 2118106 IC50 = 501.19 nM T63505 C82UBY 2130377 Ki = 50 nM T63505 CXT6M0 2180013 Ki = 130 nM T63505 C6PTI2 2192320 Ki = 272 nM T63505 C4KZ1A 2363161 Ki = 406 nM T63505 C4HW6P 2409358 IC50 = 794.33 nM T63505 CQ5I8E 2447649 Ki = 245 nM T63505 CZ35LN 2468349 IC50 = 7943.28 nM T63505 CL8K4Y 2740553 IC50 = 6309.57 nM T63505 C86LNP 2779952 IC50 > 100000 nM T63505 CV7Y5T 2807058 IC50 > 100000 nM T63505 CJ0KM7 2964715 Ki = 3474 nM T63505 C7VZO2 2964717 Ki = 845 nM T63505 C1L7AT 2964718 Ki = 170 nM T63505 CJBX04 3039851 IC50 > 100000 nM T63505 CPD6V3 3144222 Ki = 59 nM T63505 C6LO1V 3320545 Ki = 104 nM T63505 CCFI27 3320547 Ki = 44 nM T63505 CC79BS 3448811 Ki = 225 nM T63505 CCU3P7 3635406 IC50 = 380000 nM T63505 C3JTC0 3643794 Ki = 89 nM T63505 CR0DJ8 4078145 IC50 = 8000 nM T63505 C9Y7IC 4390766 Ki = 217 nM T63505 C0AY4Z 4542330 IC50 = 316.23 nM T63505 CR5I7G 4573026 Ki = 167 nM T63505 CE74CV 5059890 IC50 > 1000 nM T63505 CE1YL9 5092865 IC50 > 725000 nM T63505 C97JHC 5157299 Ki = 920 nM T63505 CR0GF5 5288018 IC50 = 17600 nM T63505 C6UL3A 5327821 IC50 = 410 nM T63505 CR3OF4 5327822 IC50 = 410 nM T63505 C9QMX2 5327823 IC50 = 1960 nM T63505 CA4G1B 5327824 IC50 = 1360 nM T63505 CY2NC3 5327825 IC50 = 1980 nM T63505 CDT07K 5327826 IC50 = 1360 nM T63505 CG36XB 5327827 IC50 = 1650 nM T63505 CF3Y6G 5327828 IC50 > 10000 nM T63505 CY1Z9E 5327829 IC50 = 150 nM T63505 CI51CH 5327830 IC50 = 3400 nM T63505 CUAW78 5327831 IC50 = 260 nM T63505 CC9US2 5327832 IC50 > 10000 nM T63505 CVGK98 5327833 IC50 = 1180 nM T63505 CGWP86 5327834 IC50 > 10000 nM T63505 C10RVD 5327835 IC50 = 6600 nM T63505 CD6B2A 5327836 IC50 > 10000 nM T63505 CY1O6K 5327837 IC50 = 3500 nM T63505 C1K8CJ 5327838 IC50 > 10000 nM T63505 CP15JO 5327839 IC50 = 3760 nM T63505 CWT9S8 5327840 IC50 = 180 nM T63505 C5EWD2 5327841 IC50 = 16500 nM T63505 C67JVQ 5327843 IC50 > 10000 nM T63505 CY23QP 5327844 IC50 = 3090 nM T63505 CN1X4Z 5327845 IC50 > 10000 nM T63505 C6TGI1 5327846 IC50 = 3600 nM T63505 CEMR07 5327847 IC50 > 10000 nM T63505 CB90GI 5327848 IC50 > 10000 nM T63505 C52MYD 5327893 IC50 = 30 nM T63505 CQ0ZP3 5327897 IC50 = 2.6 nM T63505 C7KIT4 5327898 IC50 = 5.3 nM T63505 CTC68O 5329656 IC50 > 60000 nM T63505 CUEZ35 5330437 IC50 = 490 nM T63505 CM47KI 5351344 IC50 > 10000 nM T63505 CW40OE 5574476 IC50 = 290 nM T63505 CDK3J0 5703619 IC50 = 271 nM T63505 CO9N0D 7946867 Ki = 400 nM T63505 CQ57EC 9548013 IC50 > 100000 nM T63505 CZR3M4 9799152 IC50 > 100000 nM T63505 CB9ZH4 9805421 IC50 = 2.3 nM T63505 CY3MK1 9807952 IC50 = 8.8 nM T63505 CI3O6X 9814609 IC50 = 61000 nM T63505 CX9DG5 9822042 IC50 = 20 nM T63505 C1E2DV 9826083 IC50 > 10000 nM T63505 CSH0A9 9847014 IC50 = 350 nM T63505 C3UQL7 9860872 IC50 = 34000 nM T63505 C1W4JG 9872939 IC50 = 1000 nM T63505 C5GE7T 9917045 IC50 = 480 nM T63505 CIZ13L 9943193 IC50 = 600 nM T63505 CUKH27 9943194 IC50 = 700 nM T63505 CU78NO 9947433 IC50 = 150 nM T63505 CYT7R9 9953676 IC50 = 800 nM T63505 CJ40GO 9965429 IC50 = 1500 nM T63505 CTE3K0 9982070 IC50 = 1057 nM T63505 CQZF34 9994794 IC50 > 100000 nM T63505 C26QHZ 10005638 IC50 > 10000 nM T63505 CYX27A 10006987 IC50 = 3.6 nM T63505 CA0BL8 10008474 IC50 = 7400 nM T63505 C53UTR 10022185 IC50 > 50000 nM T63505 CLI9A3 10029363 IC50 = 120 nM T63505 CMZ2S8 10029735 IC50 = 13 nM T63505 C0G5DK 10039959 IC50 = 8000 nM T63505 C54AEL 10048519 IC50 > 100000 nM T63505 CT9F2H 10053560 IC50 = 5.1 nM T63505 CUJR40 10062694 IC50 < 5 nM T63505 C6K0XB 10064040 IC50 > 50000 nM T63505 CEKL46 10070245 IC50 = 2.3 nM T63505 C2P6HN 10071040 IC50 = 22 nM T63505 C7J8YN 10073101 IC50 > 100000 nM T63505 CTAY63 10076476 IC50 = 1600 nM T63505 CFDU07 10090006 Ki = 4800 nM T63505 C8G5RH 10095463 IC50 = 5 nM T63505 C3P8WK 10110378 IC50 = 1000 nM T63505 C63CFD 10111108 IC50 = 1300 nM T63505 CL42XS 10136330 IC50 = 800 nM T63505 CUW34X 10157645 IC50 = 1900 nM T63505 CP95FO 10181075 IC50 = 6950 nM T63505 COC30E 10181160 IC50 = 200 nM T63505 CHFZ23 10266516 IC50 > 100000 nM T63505 CN51JQ 10292737 IC50 = 450 nM T63505 C7SFI1 10296883 IC50 = 3300 nM T63505 C1KFM8 10318154 IC50 = 50000 nM T63505 C27CDR 10319118 IC50 > 50000 nM T63505 C62MZJ 10320122 Ki = 7030 nM T63505 CQ80HY 10337047 IC50 > 100000 nM T63505 CET21U 10337153 IC50 > 100000 nM T63505 CUN52O 10345191 IC50 = 4.7 nM T63505 CDS29Z 10366675 IC50 = 4.8 nM T63505 CA8B5T 10390073 IC50 > 10000 nM T63505 C9RCU7 10408993 IC50 > 50000 nM T63505 CU4R9M 10413666 IC50 = 4.9 nM T63505 C7HBP6 10429593 IC50 > 10000 nM T63505 C3MI7D 10430804 IC50 > 100000 nM T63505 CSAZ29 10454329 Ki = 0.02 nM T63505 CY9DS7 10458235 IC50 = 7.6 nM T63505 C17OFQ 10476638 Ki = 260 nM T63505 CR07PO 10477008 IC50 = 70000 nM T63505 C7TJ9U 10483163 IC50 = 12 nM T63505 C78FPR 10501266 IC50 = 370 nM T63505 CJW04C 10556625 IC50 = 95900 nM T63505 CU8Q5N 10626988 IC50 = 72000 nM T63505 CNC85V 10651406 IC50 = 25700 nM T63505 CBX1F5 10674779 IC50 = 26000 nM T63505 CZP40T 10699325 IC50 = 6000 nM T63505 CU6G5Y 10708835 IC50 = 1200 nM T63505 CCN2Q5 10721885 IC50 = 46200 nM T63505 CA4FT1 10722796 IC50 = 5000 nM T63505 C0L4GE 11199718 Ki = 1200 nM T63505 CMQA73 11215316 IC50 = 12 nM T63505 CF2GE5 11222252 Ki = 370 nM T63505 CUS18W 11223073 Ki = 1500 nM T63505 CH7D3X 11233762 IC50 = 200 nM T63505 CJTP13 11280103 IC50 = 3800 nM T63505 CO2E3W 11280238 IC50 = 300 nM T63505 CBOP58 11293798 Ki > 10000 nM T63505 CE8SO6 11307464 Ki = 1.3 nM T63505 CANY24 11311217 IC50 = 1800 nM T63505 CRD9E5 11314043 IC50 = 400 nM T63505 CIL0J6 11326339 Ki = 400 nM T63505 CKY3E2 11338122 IC50 = 200 nM T63505 C26BZX 11362471 Ki > 10000 nM T63505 C3E6MX 11370613 IC50 = 50000 nM T63505 C3OCV2 11371778 IC50 = 1000 nM T63505 CWXB93 11397177 Ki > 10000 nM T63505 C3O0WI 11438191 IC50 = 5100 nM T63505 CM75ZT 11439261 Ki = 9750 nM T63505 C3EXM4 11440028 IC50 = 400 nM T63505 CFJ6B2 11441375 IC50 = 466 nM T63505 C7I6AG 11474111 IC50 = 500 nM T63505 C4Q7XD 11474276 IC50 = 110 nM T63505 C0YH2X 11478363 IC50 = 0.97 nM T63505 C3J1IY 11484016 IC50 = 20000 nM T63505 CMW72Q 11488124 IC50 = 52 nM T63505 CU18JL 11526010 Ki = 0.5 nM T63505 C20CWI 11526872 Ki = 0.3 nM T63505 CL7X4Q 11530963 IC50 = 93000 nM T63505 CTG83F 11539329 Ki > 710 nM T63505 CT64NL 11540547 IC50 = 0.43 nM T63505 CACS26 11561968 Ki > 2000 nM T63505 CJV20L 11569758 Ki = 3.5 nM T63505 CP1KN5 11577746 Ki = 0.4 nM T63505 CO9KP5 11583459 IC50 > 10000 nM T63505 CAJQ78 11584678 Ki = 3 nM T63505 CMIL86 11590363 Ki > 710 nM T63505 CF2Z5Q 11592328 Ki = 1 nM T63505 CUIW90 11599550 Ki = 2.9 nM T63505 C69FYK 11604142 Ki = 400 nM T63505 C43JZU 11604436 IC50 > 20000 nM T63505 CGU7N0 11604739 IC50 > 20000 nM T63505 C9T6SC 11640926 Ki > 710 nM T63505 CNB05F 11649873 Ki = 5.1 nM T63505 CI4A8T 11650224 IC50 = 0.43 nM T63505 CAJS96 11662893 IC50 > 20000 nM T63505 C9SL1J 11669430 Ki = 3.3 nM T63505 CKAH36 11669784 IC50 > 20000 nM T63505 C97JWR 11678625 Ki = 27 nM T63505 CU0E8O 11690457 Ki > 2000 nM T63505 CB0AP2 11705863 Ki > 10000 nM T63505 CHL5W3 11712625 Ki = 1.3 nM T63505 C7WUG6 11713575 Ki = 1.7 nM T63505 CZY05V 11719421 Ki = 11 nM T63505 CFJ4I7 11723151 IC50 = 3300 nM T63505 C9HC4M 11726643 IC50 > 100000 nM T63505 C7C2FM 11737638 IC50 = 1500 nM T63505 COX34W 11741081 Ki = 320 nM T63505 C8MOK3 11750699 IC50 < 1000 nM T63505 CP7AH3 11755812 IC50 = 14400 nM T63505 CGYV23 11779501 IC50 > 100000 nM T63505 C9JT4S 11847343 IC50 > 10000 nM T63505 CS81MP 11957378 IC50 = 68 nM T63505 C2Z8DQ 14624081 IC50 = 110000 nM T63505 C2N3WV 14638906 Ki = 500 nM T63505 CK8XF4 15209376 IC50 > 100000 nM T63505 CQN23V 15551239 IC50 > 50000 nM T63505 CHF8C5 15580688 IC50 = 1995.26 nM T63505 CXZ0O1 15858769 IC50 = 16000 nM T63505 C4I3PF 15858771 IC50 = 1700 nM T63505 C9TS5M 15950818 IC50 = 25000 nM T63505 CFPW41 16007116 Ki > 700 nM T63505 C9TU1O 16046126 IC50 > 1000 nM T63505 C3TQ4R 16099168 IC50 = 0.43 nM T63505 CQG45C 16109001 IC50 = 1280 nM T63505 CGC34R 16118737 IC50 = 2 nM T63505 C5VPH9 16129448 IC50 = 1200 nM T63505 CG68HM 16416416 IC50 = 260 nM T63505 CH4LP8 16662775 IC50 = 66 nM T63505 C6TQ2O 16664354 Ki = 2.04 nM T63505 C2IF3P 16678352 IC50 = 1960 nM T63505 C3IO1C 16679060 IC50 > 10000 nM T63505 CY1E2N 16723801 IC50 > 100000 nM T63505 CI64MP 16750094 Ki = 20 nM T63505 CL6DH1 17588993 IC50 = 11200 nM T63505 C0FC8U 17593161 IC50 = 3300 nM T63505 C97XZG 18008864 IC50 = 43.7 nM T63505 C0WEX3 19966997 IC50 > 50000 nM T63505 C97ABE 21365952 IC50 = 81.2 nM T63505 CLTH65 21365956 IC50 = 1387 nM T63505 CQK09Y 22474502 Ki = 1646 nM T63505 CBD9U4 23647620 IC50 > 50000 nM T63505 C2C3EM 23649898 IC50 = 96000 nM T63505 CML17W 23655479 Ki = 320 nM T63505 C7MT4E 23655480 Ki = 370 nM T63505 CWV5K4 23655678 Ki = 110 nM T63505 CI9PE2 23655679 Ki = 89 nM T63505 CT0SZ7 23655680 Ki = 80 nM T63505 CVW9M8 23655681 Ki = 110 nM T63505 C1MDZ7 23655682 Ki = 600 nM T63505 C10KDP 23655683 Ki = 60 nM T63505 CF3A7U 23655878 Ki = 40 nM T63505 C5TV4F 23655879 Ki = 150 nM T63505 C6JTW3 23656073 Ki = 230 nM T63505 CGIH32 23656074 Ki = 200 nM T63505 C7IU1G 23656075 Ki = 350 nM T63505 C4F1VE 23656077 Ki = 130 nM T63505 C7TG0V 23656262 Ki = 320 nM T63505 CE5XF1 23656263 Ki = 100 nM T63505 C64ESF 23656264 Ki = 250 nM T63505 CGC07X 23656265 Ki = 400 nM T63505 C8B7PK 23656266 Ki = 400 nM T63505 CN17BU 23656267 Ki = 150 nM T63505 C07QYL 23657200 IC50 = 28 nM T63505 C4JE1L 23657441 IC50 = 9.1 nM T63505 C6O8QY 23661616 Ki = 0.062 nM T63505 C2S5ZM 23661662 Ki = 44 nM T63505 C2RV3U 24180608 IC50 > 30000 nM T63505 CA3I4T 24753787 IC50 > 50000 nM T63505 C7YG1N 24759534 IC50 < 10 nM T63505 CAJ4T2 24762205 IC50 = 40 nM T63505 CQNP54 24764449 IC50 = 1000 nM T63505 C0EKO5 24772654 IC50 = 0.4 nM T63505 CP9G0L 24783392 IC50 = 1900 nM T63505 CB9N8E 24802574 Ki = 80 nM T63505 CQK54U 24807247 Ki = 730 nM T63505 C91MSB 24807248 Ki = 440 nM T63505 CF39RQ 24807249 Ki = 200 nM T63505 C5CXU0 24807250 Ki = 100 nM T63505 CYVE35 24807251 Ki = 20 nM T63505 C5GW2A 24807252 Ki = 120 nM T63505 CBD73X 24807440 Ki = 200 nM T63505 CYV8G5 24807442 Ki = 80 nM T63505 C1B8AS 24807618 Ki = 2000 nM T63505 CS6DA5 24807619 Ki = 40 nM T63505 CW0G8H 24812719 IC50 = 1400 nM T63505 CCP2M3 24822704 IC50 > 50000 nM T63505 CX94DT 24823073 Ki = 42 nM T63505 CG0K1Z 24824046 IC50 = 240 nM T63505 CJ0CU5 24825841 IC50 = 0.4 nM T63505 CSO9H2 24826558 IC50 = 2.3 nM T63505 C7R2YB 24826632 IC50 = 26 nM T63505 CBVE95 24826654 IC50 = 2.3 nM T63505 C5M9GS 24826656 IC50 = 9.1 nM T63505 CR5A6Y 24826712 IC50 = 45 nM T63505 CE9VG3 24826714 IC50 = 6.4 nM T63505 C1YH5C 24826733 IC50 = 26 nM T63505 CDR74A 24826736 IC50 = 13 nM T63505 CURN06 24826798 IC50 = 15 nM T63505 CV3R8D 24826800 IC50 = 2.4 nM T63505 C1D3US 24826801 IC50 = 5.3 nM T63505 CGTP30 24826816 IC50 = 49 nM T63505 CF5SQ7 24826817 IC50 = 22 nM T63505 CUM6E0 24826878 IC50 = 31 nM T63505 CXV63D 24826879 IC50 = 12 nM T63505 CKQ68M 24826880 IC50 = 2.3 nM T63505 CL3FM9 24826893 IC50 = 15 nM T63505 CKM84D 24826896 IC50 = 24 nM T63505 CB2FQ3 24826975 IC50 = 14 nM T63505 CAD94Z 24827068 IC50 = 1.4 nM T63505 CH71YI 24827072 IC50 = 56 nM T63505 CVUB20 24827163 IC50 = 19 nM T63505 C2BCG1 24827164 IC50 = 23 nM T63505 C36RQD 24862886 IC50 = 3.6 nM T63505 C83FEO 24863033 IC50 = 129 nM T63505 CWR58K 24863036 IC50 = 29 nM T63505 CUZ7O0 24863123 IC50 = 3.6 nM T63505 CC8OF2 24871562 IC50 = 62.7 nM T63505 CDJE41 24879368 IC50 > 25000 nM T63505 CFK2B9 24882503 IC50 = 250 nM T63505 C43HWQ 24883287 IC50 = 500 nM T63505 C8DA5Q 24883334 IC50 < 100 nM T63505 CY8L7E 24896769 IC50 > 10000 nM T63505 CB79YC 24905143 IC50 = 70 nM T63505 C2DC9J 24905144 IC50 = 1200 nM T63505 CN6V8Z 24905145 IC50 = 1 nM T63505 CSB7P5 24905148 IC50 = 1400 nM T63505 CGSF21 24905149 IC50 = 17000 nM T63505 CVDG02 24905150 IC50 < 1 nM T63505 CWH6C5 24905152 IC50 = 140 nM T63505 C0HE2Q 24905153 IC50 = 170 nM T63505 C7QSC9 24905154 IC50 = 3200 nM T63505 CO9D0K 24905155 IC50 = 2000 nM T63505 C5W9UR 24905157 IC50 = 2600 nM T63505 CC1DA3 24905158 IC50 = 4500 nM T63505 COW79F 24905159 IC50 = 13000 nM T63505 CFPA53 24905160 IC50 = 17000 nM T63505 C2O0JX 24905161 IC50 = 11000 nM T63505 CA72BE 24905162 IC50 = 11000 nM T63505 CQN6X9 24905163 IC50 = 50000 nM T63505 CD4O1F 24905165 IC50 = 13000 nM T63505 CKL48T 24905166 IC50 = 7900 nM T63505 C76VYL 24905167 IC50 = 50000 nM T63505 C7K5PU 24905168 IC50 = 3600 nM T63505 CZ57ID 24905169 IC50 = 1700 nM T63505 C2DHX9 24905170 IC50 = 32000 nM T63505 CSB96E 24905171 IC50 = 50000 nM T63505 CWZ0R2 24905172 IC50 = 1300 nM T63505 CY3B6M 24905175 IC50 = 558 nM T63505 CW7UA3 24905176 IC50 = 2500 nM T63505 CW1V0H 24905177 IC50 = 830 nM T63505 CO6Y0L 24905178 IC50 = 11200 nM T63505 C60NQW 24905179 IC50 = 1190 nM T63505 C4MO8B 24905180 IC50 = 75 nM T63505 COJI47 24905181 IC50 = 63 nM T63505 CS0B2C 24905182 IC50 = 24 nM T63505 C1H4BT 24905183 IC50 = 26 nM T63505 C4WHK9 24905184 IC50 = 1500 nM T63505 C7Q4MZ 24905185 IC50 = 527 nM T63505 CS4IP1 24905186 IC50 = 26 nM T63505 C69QWO 24905187 IC50 = 920 nM T63505 C85ANB 24905188 IC50 = 295 nM T63505 CNHD75 24905189 IC50 = 1000 nM T63505 C9JUO2 24905190 IC50 = 2600 nM T63505 CPR03K 24905191 IC50 = 2200 nM T63505 CTAG19 24905193 IC50 = 234 nM T63505 C7VJM5 24905194 IC50 = 5200 nM T63505 CEP1L3 24905195 IC50 = 538 nM T63505 CP68ZD 24905196 IC50 = 893 nM T63505 C8Z0RJ 24905197 IC50 = 608 nM T63505 CN9RT0 24905198 IC50 = 8700 nM T63505 CHI78P 24905200 IC50 = 1000 nM T63505 CO6PE8 24905201 IC50 = 200 nM T63505 CZ63HS 24905202 IC50 = 22 nM T63505 C2X0FC 24905203 IC50 = 110 nM T63505 C0WCE3 24905204 IC50 = 100000 nM T63505 CNK50B 24905205 IC50 = 1500 nM T63505 C12DPB 24905206 IC50 = 140 nM T63505 C8N0RH 24905207 IC50 = 15000 nM T63505 CYA5G2 24905208 IC50 = 5100 nM T63505 CDV2B4 24905209 IC50 = 1500 nM T63505 CEFK68 24905210 IC50 = 310 nM T63505 CUFP12 24905211 IC50 = 759 nM T63505 C0JG8L 24905212 IC50 = 165 nM T63505 CQ13ZI 24905215 IC50 = 12000 nM T63505 C6VI8F 24905216 IC50 = 3800 nM T63505 CXNH25 24905217 IC50 = 2100 nM T63505 C2PN9S 24905218 IC50 = 2200 nM T63505 C9O2AL 24905219 IC50 = 4300 nM T63505 CIT7U8 24905220 IC50 = 2000 nM T63505 CMD26S 24905221 IC50 = 690 nM T63505 C4R8WC 24905222 IC50 = 816 nM T63505 C47SHA 24905223 IC50 = 498 nM T63505 C1DY2R 24905224 IC50 = 469 nM T63505 CS0XF9 24905225 IC50 = 2000 nM T63505 CG5VX2 24905226 IC50 = 35000 nM T63505 C57QEO 24905227 IC50 = 100000 nM T63505 C7CG5E 24905228 IC50 = 3000 nM T63505 CHP5D1 24905229 IC50 = 2200 nM T63505 CXP09S 24905230 IC50 = 2000 nM T63505 CY7XG1 24905231 IC50 = 65000 nM T63505 C7JFQ2 24905232 IC50 = 2000 nM T63505 C2JM1P 24905233 IC50 = 6400 nM T63505 CC3BF0 24905234 IC50 = 100000 nM T63505 CE57FI 24905235 IC50 = 1300 nM T63505 CUP20O 24905236 IC50 = 3400 nM T63505 CLC6Q2 24905237 IC50 = 5000 nM T63505 C9M1GI 24905238 IC50 = 688 nM T63505 CVD72F 24905239 IC50 = 327 nM T63505 CK38IZ 24905240 IC50 = 1100 nM T63505 CO2V5E 24905241 IC50 = 8400 nM T63505 CZBA19 24905244 IC50 = 87 nM T63505 CQ8OI1 24905246 IC50 = 14000 nM T63505 CIF2J5 24905251 IC50 = 260 nM T63505 CPTE58 24905252 IC50 = 208 nM T63505 C6XHJ7 24905272 Ki = 69 nM T63505 CP50RD 24905280 IC50 = 14 nM T63505 CG13ZM 24905281 IC50 = 113 nM T63505 CF0S6X 24905282 IC50 = 2100 nM T63505 C5HBL0 24905284 IC50 = 13000 nM T63505 C2Z5DN 24905285 IC50 = 560 nM T63505 CL6GH8 24905286 IC50 = 784 nM T63505 CKYO98 24905287 IC50 = 31 nM T63505 CRNQ65 24905288 IC50 = 90 nM T63505 COD7I5 24905289 IC50 = 160 nM T63505 C4LP7E 24905290 IC50 = 233 nM T63505 CE9JC2 24905291 IC50 = 530 nM T63505 C2GI1R 24905292 IC50 = 6150 nM T63505 CHW8C4 24905293 IC50 = 177 nM T63505 CQF0H1 24905294 IC50 = 56 nM T63505 CNO7X0 24905295 IC50 = 5.5 nM T63505 C5WRG7 24905296 IC50 = 850 nM T63505 CQ1S0U 24905297 IC50 = 14600 nM T63505 C4UES7 24905298 IC50 = 6050 nM T63505 CMS69P 24905299 IC50 = 7930 nM T63505 CC0U5M 24905300 IC50 = 1.2 nM T63505 CW7X6S 24905301 IC50 = 5842 nM T63505 C97IQV 24905302 IC50 = 4.3 nM T63505 CSJ47V 24905303 IC50 = 4500 nM T63505 CPN74C 24905304 IC50 = 1044 nM T63505 C5CS3N 24905305 IC50 = 82 nM T63505 CK4XE9 24905307 IC50 = 393 nM T63505 CTU6Z3 24905308 IC50 = 565 nM T63505 C9SQX1 24905309 IC50 = 72 nM T63505 CM75JP 24905310 IC50 = 483 nM T63505 C9Q2BJ 24905311 IC50 = 2050 nM T63505 C9VUA1 24905312 IC50 = 505 nM T63505 CU3RS1 24905313 IC50 = 4000 nM T63505 CYG3H2 24905314 IC50 = 293 nM T63505 CV5Q7O 24905315 IC50 = 6.4 nM T63505 C8SA3O 24905316 IC50 = 68 nM T63505 CI5MN3 24905317 IC50 = 21 nM T63505 CJ1P7K 24905318 IC50 = 17 nM T63505 C1T6YQ 24905319 IC50 = 21 nM T63505 CAU86X 24905320 IC50 = 21 nM T63505 C54ISY 24905321 IC50 = 199 nM T63505 C2GE5I 24905322 IC50 = 130 nM T63505 C8D6YK 24905323 IC50 = 726 nM T63505 C5NZH9 24905324 IC50 = 695 nM T63505 C9D6JR 24905325 IC50 = 55 nM T63505 CLZT41 24905326 IC50 = 32 nM T63505 CW8FD3 24905327 IC50 = 67 nM T63505 CHB7A2 24905328 IC50 = 963 nM T63505 CA8EI3 24905329 IC50 = 433 nM T63505 CCQ0O7 24905330 IC50 = 4400 nM T63505 CJ81AS 24905331 IC50 = 109 nM T63505 C8PW4H 24905332 IC50 = 23 nM T63505 C2Y5TF 24905333 IC50 = 45 nM T63505 CH9FL5 24905334 IC50 = 6400 nM T63505 C1S0PC 24905335 IC50 = 12000 nM T63505 C8N9MV 24905336 IC50 = 319 nM T63505 C9E8BJ 24905338 IC50 = 58000 nM T63505 CX85AC 24905341 IC50 = 50000 nM T63505 CKZ80E 24905342 IC50 = 52 nM T63505 CO8SH1 24905343 IC50 = 4100 nM T63505 C7IZL6 24905344 IC50 = 1800 nM T63505 C4EG8R 24993189 IC50 > 10000 nM T63505 CB38WD 25027538 IC50 = 1760 nM T63505 C7GHJ8 25028631 IC50 > 0.4 ug.mL-1 T63505 C2ICS7 25065806 IC50 = 3.58 nM T63505 CQ1E0N 25185128 Ki = 340 nM T63505 CP3EN4 25185129 Ki = 200 nM T63505 CYN31L 25185130 Ki = 220 nM T63505 C40LQJ 25185131 Ki = 400 nM T63505 C2PR9C 25185132 Ki = 390 nM T63505 CF8GX1 25185133 Ki = 300 nM T63505 CE4LB1 25185134 Ki = 500 nM T63505 CUVP43 25185398 Ki = 250 nM T63505 CH8J4V 25185399 Ki = 520 nM T63505 COL73S 25185400 Ki = 100 nM T63505 CP6G0U 25185403 Ki = 320 nM T63505 C3FU2E 25185404 Ki = 1400 nM T63505 CZ80GV 25185687 Ki = 970 nM T63505 CIU1P5 25185688 Ki = 190 nM T63505 CXQ10W 25185691 Ki = 320 nM T63505 CZ60BO 25185692 Ki = 160 nM T63505 CXMN65 25185693 Ki = 330 nM T63505 C4L2VA 25185968 Ki = 280 nM T63505 C1LIZ0 25185969 Ki = 880 nM T63505 C81UNB 25185970 Ki = 550 nM T63505 CX2IE4 25185971 Ki = 880 nM T63505 C94EPM 25185972 Ki = 270 nM T63505 CH3X8S 25185973 Ki = 280 nM T63505 CZG39U 25189269 Ki = 400 nM T63505 CPZ70U 25189270 Ki = 570 nM T63505 CF6GK9 25189271 Ki = 110 nM T63505 C4QG2L 25189272 Ki = 970 nM T63505 C7FMJ5 25189273 Ki = 220 nM T63505 CT5WQ7 25195368 IC50 = 33 nM T63505 CNG96H 25210579 IC50 > 10000 nM T63505 C6L9FV 25211674 IC50 = 17.3 nM T63505 C3F7QN 25211675 IC50 = 2.77 nM T63505 C43UPC 25211772 IC50 = 15.8 nM T63505 CC71QJ 27666048 IC50 = 5600 nM T63505 C5BO1L 40544927 IC50 = 310 nM T63505 CIW8V3 40833444 Ki = 369 nM T63505 CVM13K 42596931 IC50 = 24 nM T63505 CU53WB 42596953 IC50 = 5300 nM T63505 CAG14D 42609923 IC50 = 290 nM T63505 C7GIQ3 42625508 IC50 = 9200 nM T63505 CVZ83M 42625582 IC50 = 1120 nM T63505 C5MD9E 42625892 IC50 = 34000 nM T63505 CI9DK5 42628614 IC50 = 7900 nM T63505 CKG80R 42805643 Ki = 195 nM T63505 CLW80F 44160269 IC50 = 3400 nM T63505 CWT68J 44186427 IC50 = 141 nM T63505 CCFQ29 44187005 IC50 = 286 nM T63505 CN4FS2 44195235 IC50 = 79.8 nM T63505 CK73NR 44219749 IC50 > 50000 nM T63505 C1OJ5W 44221514 IC50 = 74000 nM T63505 C48QGV 44221515 IC50 = 9900 nM T63505 CWB74L 44221727 IC50 = 157000 nM T63505 CK5G4H 44221730 IC50 = 236000 nM T63505 C4H6WC 44221731 IC50 = 60000 nM T63505 CP3Z1S 44221732 IC50 = 146000 nM T63505 C2K5IO 44221929 IC50 = 48 nM T63505 C9LU0Y 44221931 IC50 = 37000 nM T63505 CB2A0O 44222109 IC50 = 243000 nM T63505 CXKZ46 44222110 IC50 = 26000 nM T63505 C4YS1K 44222111 IC50 = 40000 nM T63505 C54QWZ 44222112 IC50 = 5700 nM T63505 CV8P4L 44222285 IC50 = 23000 nM T63505 C7NK8F 44222286 IC50 = 59000 nM T63505 C42AML 44222458 IC50 = 267000 nM T63505 CK3S2I 44222459 IC50 = 23000 nM T63505 CJ43YR 44222636 IC50 = 62000 nM T63505 C65TLI 44222639 IC50 = 542 nM T63505 CY5IU1 44222822 IC50 = 72000 nM T63505 C2MJI4 44222823 IC50 = 24000 nM T63505 C6MPO3 44222824 IC50 = 38 nM T63505 CMRX16 44273620 IC50 = 5800 nM T63505 CCH89M 44300026 IC50 = 2000 nM T63505 CV5QH7 44300064 IC50 = 1200 nM T63505 CTJV27 44300144 IC50 = 4900 nM T63505 CVD6B1 44300175 IC50 = 22000 nM T63505 CA2HD0 44300205 IC50 = 1200 nM T63505 CJQ1T0 44300215 IC50 = 100000 nM T63505 CBGM82 44300226 IC50 = 17000 nM T63505 C9FX3G 44300234 IC50 = 14000 nM T63505 CY6P9K 44318047 IC50 > 100000 nM T63505 C92TBJ 44324648 IC50 = 15300 nM T63505 CY0XF5 44340726 IC50 > 10000 nM T63505 C0KD4U 44346053 IC50 > 10000 nM T63505 CYV2D7 44368815 IC50 = 5330 nM T63505 C0BSN4 44383430 IC50 = 94 nM T63505 C2F7SL 44395745 IC50 = 930 nM T63505 CP3LJ6 44395749 IC50 = 870 nM T63505 CZR42M 44395763 IC50 = 56 nM T63505 C5P6LS 44395789 IC50 = 175 nM T63505 CEYC94 44395793 IC50 = 1000 nM T63505 CU9XQ0 44395880 IC50 > 5000 nM T63505 CYF8U6 44395904 IC50 = 280 nM T63505 C5DR6W 44395926 IC50 > 3400 nM T63505 CLE93Z 44425266 Ki = 16 nM T63505 CHA07Y 44425863 IC50 = 220 nM T63505 CICY26 44425865 IC50 = 3110 nM T63505 CV3AQ9 44425866 IC50 > 10000 nM T63505 CGOU30 44425867 IC50 = 156 nM T63505 CVR96G 44425868 IC50 = 18 nM T63505 C2ZBH4 44425870 IC50 = 33 nM T63505 CZE2S4 44425871 IC50 = 180 nM T63505 CEX4Q9 44430662 IC50 = 32 nM T63505 CYB28E 44430665 IC50 = 140 nM T63505 C5ZKI8 44435586 Ki = 240 nM T63505 C5R4QE 44442729 Ki = 950 nM T63505 CGC76I 44442730 Ki > 10000 nM T63505 CJM6N5 44442731 Ki > 10000 nM T63505 CH2FS6 44442732 Ki > 10000 nM T63505 CZ7FC6 44442733 Ki > 10000 nM T63505 C6PNZ4 44442734 Ki = 1800 nM T63505 C8N1EQ 44442735 Ki = 1800 nM T63505 C26EVP 44442736 Ki = 300 nM T63505 C0S6PN 44442737 Ki = 390 nM T63505 CAZ5O7 44442738 Ki = 200 nM T63505 CM9XW1 44442739 Ki > 10000 nM T63505 CFOH51 44442740 Ki > 10000 nM T63505 CX10DZ 44442742 Ki = 770 nM T63505 CN12IA 44442744 Ki > 10000 nM T63505 C0DOP6 44442745 Ki = 300 nM T63505 C6N4KQ 44444040 Ki = 2.6 nM T63505 C1L6MG 44444041 Ki = 1.7 nM T63505 CJ49DR 44444043 Ki = 4.2 nM T63505 CWD69U 44444045 Ki = 7.7 nM T63505 C90DMA 44444053 Ki = 4.4 nM T63505 C3DI2R 44444055 Ki = 3.5 nM T63505 CBY1F9 44444057 Ki = 3.4 nM T63505 CZ27CI 44444060 Ki = 24 nM T63505 CBU8P5 44454498 Ki = 73 nM T63505 C0ZL8E 44454721 Ki = 1260 nM T63505 C3RY8Z 44454722 Ki = 760 nM T63505 C2KJO6 44454776 Ki = 210 nM T63505 CA2JO0 44454803 Ki = 189 nM T63505 CH64KP 44454904 Ki = 92 nM T63505 C6CQJ0 44454939 Ki = 83 nM T63505 C30NZA 44475985 IC50 = 8 nM T63505 CV9Z6W 44517648 IC50 < 0.46 nM T63505 C4WRN5 44541014 IC50 = 9.7 nM T63505 C3VRO9 44557921 IC50 > 10000 nM T63505 CQL6U3 44561590 IC50 = 5.93 nM T63505 CFS16E 44561591 IC50 = 54.3 nM T63505 CCVU76 44561592 IC50 = 73.3 nM T63505 C4QBE6 44561593 IC50 = 626 nM T63505 CEF4G0 44561735 IC50 = 69.4 nM T63505 CR87GD 44561736 IC50 = 16.7 nM T63505 CA25TK 44561737 IC50 = 2.36 nM T63505 C8TRZ9 44561787 IC50 = 17.6 nM T63505 C7YK5F 44561788 IC50 = 19.5 nM T63505 CDK0X8 44561828 IC50 = 3.02 nM T63505 C38YGU 44561829 IC50 = 6.8 nM T63505 C28NDO 44561830 IC50 = 1.63 nM T63505 C4C6VA 44561831 IC50 = 1.8 nM T63505 CJ73WK 44561866 IC50 = 7.32 nM T63505 CMKB42 44561867 IC50 = 1.57 nM T63505 C1TQ2I 44561868 IC50 < 0.46 nM T63505 C6MA5F 44561869 IC50 = 0.5 nM T63505 CDVC07 44561908 IC50 = 32.3 nM T63505 CLB68G 44561909 IC50 < 0.46 nM T63505 CL87KN 44564189 IC50 = 820 nM T63505 C1X9JM 44564254 IC50 > 0.4 ug.mL-1 T63505 CMQ1Y9 44564255 IC50 > 0.4 ug.mL-1 T63505 CS43ER 44564256 IC50 > 0.4 ug.mL-1 T63505 CC4UD7 44564257 IC50 > 0.4 ug.mL-1 T63505 C3HW7L 44570553 IC50 > 30000 nM T63505 C17PVE 44570554 IC50 > 30000 nM T63505 CLOY92 44570599 IC50 = 300 nM T63505 CK06LT 44570600 IC50 = 4000 nM T63505 COM65J 44572384 IC50 > 100000 nM T63505 CV91YE 44572385 IC50 = 4100 nM T63505 C3CB2K 44572429 IC50 = 31000 nM T63505 CM2Q8J 44572430 IC50 = 22000 nM T63505 CAN4B0 44572431 IC50 = 7800 nM T63505 CMAT21 44572489 IC50 = 39000 nM T63505 CU1SY9 44572490 IC50 = 14000 nM T63505 CSD74G 44572491 IC50 = 10000 nM T63505 CA9WO3 44572537 IC50 = 35000 nM T63505 C06SLW 44572538 IC50 = 24000 nM T63505 CY8TG3 44572539 IC50 = 8500 nM T63505 C1JR4C 44572540 IC50 = 17000 nM T63505 CZ0PA9 44572581 IC50 = 8800 nM T63505 CD9VR5 44572582 IC50 = 4000 nM T63505 CG5UK0 44572584 IC50 = 2000 nM T63505 CMX32U 44572633 IC50 = 1700 nM T63505 CMZ57P 44576263 IC50 < 5 nM T63505 CP80CQ 44578359 Ki = 791 nM T63505 C28QLM 44605035 IC50 > 50000 nM T63505 C75XHS 44605037 IC50 > 50000 nM T63505 CU3RF1 45139989 IC50 > 10000 nM T63505 CQGZ06 45139991 IC50 > 10000 nM T63505 CZC5V0 45272013 Ki = 300 nM T63505 CA06GW 45487959 IC50 = 12 nM T63505 CUMF37 45487992 IC50 = 8.2 nM T63505 CFE79C 45487997 IC50 = 1.4 nM T63505 C96BNW 46179972 IC50 = 5 nM T63505 CF57GK 46215462 IC50 > 700 nM T63505 CY3HW5 46224684 IC50 > 10000 nM T63505 C1J6GR 46224908 IC50 > 10000 nM T63505 CYT37A 46232443 IC50 > 50000 nM T63505 C48ZVW 46232555 IC50 = 10000 nM T63505 CS9B1U 46232556 IC50 > 50000 nM T63505 C85RJI 46233108 IC50 = 17000 nM T63505 C19SZF 46233185 IC50 > 50000 nM T63505 C7ON5A 46233287 IC50 > 10000 nM T63505 C1S4LH 46398810 IC50 = 80 nM T63505 C2Q9UH 46837263 IC50 = 19 nM T63505 C5P7IT 46837264 IC50 = 19 nM T63505 C0VG9W 46837265 IC50 = 54 nM T63505 C2YT9M 46837380 IC50 = 14 nM T63505 C4MO7P 46838615 IC50 = 30 nM T63505 CL07DO 46838818 IC50 > 150000 nM T63505 CNW6I7 46838966 IC50 = 290 nM T63505 C9DR6V 46838967 IC50 = 60000 nM T63505 C1ZQ8P 46839048 IC50 = 9 nM T63505 CSCI52 46839177 IC50 = 78 nM T63505 C3D7LM 46839179 IC50 = 19 nM T63505 C1OZX4 46839180 IC50 = 18 nM T63505 CRU71E 46839181 IC50 = 6.9 nM T63505 C1CVI7 46839312 IC50 = 42 nM T63505 CGU61T 46839313 IC50 = 69 nM T63505 C2E7HI 46839314 IC50 = 41 nM T63505 CZC6U5 46839315 IC50 = 42 nM T63505 C0QOJ6 46844437 Ki = 700 nM T63505 C8Q5MT 46861577 IC50 = 709 nM T63505 C1YW2Q 46866422 IC50 = 460 nM T63505 C9LI2B 46866423 IC50 = 184 nM T63505 CP68SD 46866425 IC50 = 654 nM T63505 C7FG5S 46866426 IC50 = 2300 nM T63505 CO3P0J 46866604 IC50 < 50000 nM T63505 CJOM49 46880136 IC50 = 563 nM T63505 C67UEP 46881960 IC50 = 25 nM T63505 C0WYM1 46898022 IC50 = 6000 nM T63505 CWM9H3 46900076 IC50 < 5 nM T63505 CRXG74 46911674 IC50 = 240 nM T63505 C60GAV 46929544 IC50 = 503 nM T63505 CP34VL 46929748 IC50 > 1000 nM T63505 CCN08S 46934144 IC50 > 100000 nM T63505 C0E2DY 46934424 Ki = 70 nM T63505 C1QR2X 46934425 Ki = 8 nM T63505 CUIX25 49766392 IC50 = 6200 nM T63505 C2Z6HW 49797814 IC50 = 300 nM T63505 CBHE98 49797871 IC50 = 440 nM T63505 CJE0I4 49798770 IC50 = 23 nM T63505 CL3M5D 49798776 IC50 = 28 nM T63505 C9V3TO 49798958 IC50 = 1.6 nM T63505 CHSF07 49806372 IC50 > 1000 nM T63505 C5ME3S 49806721 IC50 > 50000 nM T63505 CF91RS 49843531 IC50 > 10000 nM T63505 CG32IB 49850407 Ki = 750 nM T63505 C8EOD9 49850435 Ki = 1600 nM T63505 CE7D2J 49855568 IC50 = 7700 nM T63505 CFD9P3 49855569 IC50 = 2700 nM T63505 C1AU5N 49855758 IC50 = 4900 nM T63505 CIFK93 49855759 IC50 = 4500 nM T63505 CK48OJ 49855760 IC50 = 6000 nM T63505 CZI3M1 49855761 IC50 = 4900 nM T63505 CRPZ58 49855949 IC50 = 2900 nM T63505 CTU0K3 49855950 IC50 = 4900 nM T63505 CF85NL 49855951 IC50 = 6900 nM T63505 CF7YS9 49855952 IC50 = 1700 nM T63505 CJU38G 49855953 IC50 = 1700 nM T63505 CF6L5C 49863824 IC50 < 10 nM T63505 C67NRO 49865422 Ki = 60 nM T63505 CM2FW0 49865465 Ki = 2000 nM T63505 C58JGI 49865466 Ki = 40 nM T63505 CK4UA2 49865467 Ki = 40 nM T63505 C75OVG 49865512 Ki = 900 nM T63505 CHM90X 49865513 Ki = 20 nM T63505 CGUX26 49865514 Ki = 20 nM T63505 C78ATS 49865565 Ki = 0.02 nM T63505 CD2K4R 50908681 IC50 = 392000 nM T63505 C61DVY 50990961 IC50 = 1.2 nM T63505 CV3UP9 50992247 IC50 < 0.5 nM T63505 CS9G6E 50997096 IC50 > 10000 nM T63505 CSC61J 51037611 IC50 = 49.7 nM T63505 CU1L3G 51038269 IC50 = 0.34 nM T63505 C46STW 51346068 Ki > 1250000 nM T63505 CB9C8G 51351016 IC50 > 20000 nM T63505 COD9Y2 51351017 IC50 > 20000 nM T63505 CW96FU 51351018 IC50 > 20000 nM T63505 CR9T2E 51351019 IC50 > 20000 nM T63505 CG5IK8 52936268 IC50 > 100000 nM T63505 CEQN27 52936621 Ki > 1000 nM T63505 CU1P2L 52940797 IC50 = 65000 nM T63505 CDHJ08 52942235 IC50 = 50000 nM T63505 C1XEV2 52943394 IC50 = 1280 nM T63505 CWPC54 52945348 IC50 = 12000 nM T63505 C4NLX7 52945630 IC50 = 6000 nM T63505 CXD6T8 52945845 IC50 = 16000 nM T63505 CHJS47 52951432 Ki = 390 nM T63505 CY6JF8 52951435 Ki = 2000 nM T63505 CE03RQ 52951437 Ki = 720 nM T63505 C4LDA0 52951544 Ki = 220 nM T63505 C9UH8Q 52951545 Ki = 340 nM T63505 C0LTS2 52951546 Ki = 90 nM T63505 C2MVU5 52951547 Ki = 580 nM T63505 CFY9W7 52951548 Ki = 270 nM T63505 CY7W0Z 52951664 Ki = 120 nM T63505 CBI6V7 52951665 Ki = 150 nM T63505 C93XNY 52951666 Ki = 1600 nM T63505 CJ7UC0 52951667 Ki = 2100 nM T63505 CE5YZ0 52951668 Ki = 660 nM T63505 C9OX0Z 52951669 Ki = 1200 nM T63505 C2CT5J 53236670 IC50 = 6050 nM T63505 C3M6LV 53236671 IC50 > 100000 nM T63505 CZ5L6F 53239373 IC50 = 20840 nM T63505 C2WFI8 53239374 IC50 > 100000 nM T63505 C0ZHF8 53239375 IC50 > 100000 nM T63505 CD1EQ3 53239587 IC50 > 100000 nM T63505 C09SDH 53257410 IC50 > 10000 nM T63505 CU95KZ 53316738 Ki = 64 nM T63505 C2W9OA 53324451 IC50 > 10000 nM T63505 CNPM14 53341082 IC50 > 3000 nM T63505 C9D0TP 53346431 Ki > 15000 nM T63505 C0SWH5 53348216 IC50 > 40000 nM T63505 CM7P3W 53357328 IC50 = 370 nM T63505 CBK9Q6 53357848 IC50 > 10000 nM T63505 C8NA4L 53384644 IC50 > 30000 nM T63505 CW06MH 54581358 IC50 = 17.4 nM T63505 CSD8K1 54582383 IC50 = 55 nM T63505 CCFX61 54582384 IC50 = 4.3 nM T63505 C95EWX 54583367 IC50 = 72.6 nM T63505 CY4O2I 54584313 IC50 = 40.3 nM T63505 CX41MJ 54584314 IC50 = 18 nM T63505 C0E6DP 54585283 IC50 = 28.6 nM T63505 C57MIX 54585284 IC50 = 48.7 nM T63505 C1R2MN 54586231 IC50 = 1000 nM T63505 C7AUH4 54586232 IC50 = 12 nM T63505 C72MJD 54587257 IC50 = 4.8 nM T63505 CE1ZK6 54759168 IC50 > 10000 nM T63505 C8AB1J 54759606 Ki = 120 nM T63505 C6TN0K 54764678 IC50 = 1100 nM T63505 CM6EV1 54764680 IC50 > 25000 nM T63505 C9EMO2 54765177 IC50 = 285 nM T63505 CM8JX1 56604907 IC50 = 10 nM T63505 C9DX3J 56649281 IC50 = 53.32 nM T63505 CA51VH 56662318 Ki = 1000 nM T63505 C1MUS9 56662319 Ki = 1860 nM T63505 C3B6TD 56662320 Ki = 770 nM T63505 C0QFK5 56679360 Ki = 4920 nM T63505 C0UI3E 56682663 Ki = 1070 nM T63505 CBOD63 56835089 IC50 > 30000 nM T63505 CC06BM 56835765 Ki > 10000 nM T63505 CLNY43 56835766 Ki > 10000 nM T63505 CCR71V 56835771 Ki = 5500 nM T63505 CR16SD 56947170 IC50 = 1110 nM T63505 CJ47MX 56963907 IC50 > 10000 nM T63505 C9L6FD 56963908 IC50 = 4600 nM T63505 CE50IB 56963909 IC50 > 10000 nM T63505 CI6QE5 56970263 IC50 < 500 nM T63505 CPHX64 57325478 IC50 > 50000 nM T63505 CQ9BW4 57325479 IC50 > 50000 nM T63505 C1JLW8 57332840 IC50 = 2160 nM T63505 CD01JZ 57332841 IC50 = 5270 nM T63505 CCFK37 57332844 IC50 = 2270 nM T63505 CK1SR7 57332969 IC50 = 2490 nM T63505 C5TRE2 57332970 IC50 = 1370 nM T63505 C46TJK 57332974 IC50 = 6840 nM T63505 C09ZJY 57333095 IC50 = 7710 nM T63505 CKVG97 57394105 IC50 < 1000 nM T63505 CE1A9V 57394653 IC50 = 109 nM T63505 CD6Y9Z 57395116 IC50 > 30000 nM T63505 C8W6IG 57395117 IC50 > 30000 nM T63505 CG7S0D 57396882 IC50 > 30000 nM T63505 C4J6UZ 57397845 IC50 < 1000 nM T63505 CF3HI1 57523419 IC50 = 390 nM T63505 CS75LF 57659335 IC50 = 430 nM T63505 CVK0G4 58056356 IC50 > 50000 nM T63505 CH7L5N 58172700 IC50 = 135.8 nM T63505 C4V7FY 58191950 IC50 = 15000 nM T63505 CPCA29 58191961 IC50 = 27000 nM T63505 C7HF1L 58191965 IC50 = 7000 nM T63505 C8LWY9 58191997 IC50 = 11000 nM T63505 C6BPR2 58985201 IC50 > 30000 nM T63505 CT3EW2 59292007 IC50 > 1000 nM T63505 CXJ63M 59603829 IC50 < 10 nM T63505 CQEU96 59603842 IC50 = 1.3 nM T63505 C1MR8Q 60097495 IC50 > 1000 nM T63505 CA0LN1 60202314 IC50 = 1170 nM T63505 CS1WL6 60202315 IC50 = 176 nM T63505 C7SGT6 60202316 IC50 = 40 nM T63505 CU79HD 60202383 IC50 = 51 nM T63505 C6D2XK 60340072 IC50 = 12589.25 nM T63505 CCT79I 60581473 IC50 = 2511.89 nM T63505 C9ZCT2 62705065 IC50 > 1000 nM T63505 CUBL90 66545750 IC50 = 864 nM T63505 CD2BZ5 66549796 IC50 = 610 nM T63505 CK6WO0 66552478 IC50 < 10000 nM T63505 C3DG4W 66552583 IC50 = 100 nM T63505 C3SQ4B 66552584 IC50 = 10 nM T63505 CI3J2H 66552648 IC50 = 550 nM T63505 CA9Z7N 66552722 IC50 > 10000 nM T63505 CT6D3Y 66552723 IC50 > 10000 nM T63505 C2DL4Q 66552781 IC50 > 10000 nM T63505 CXB5R0 66552850 IC50 > 10000 nM T63505 C10AMI 66553589 IC50 = 4990 nM T63505 C9QF6B 66559005 IC50 = 56 nM T63505 CQK4Y2 66570958 IC50 = 480 nM T63505 C5RAC8 66571005 IC50 = 700 nM T63505 C5UFY3 66571008 IC50 = 210 nM T63505 C20EXP 66571075 IC50 = 1100 nM T63505 C3WF4H 66571076 IC50 = 760 nM T63505 CYS96O 66571078 IC50 = 3070 nM T63505 CPW01U 66571135 IC50 = 320 nM T63505 CC04XH 66571138 IC50 = 480 nM T63505 CJL68E 66571195 IC50 > 3000 nM T63505 CYFL93 66571254 IC50 > 3000 nM T63505 C3WM6R 66571316 IC50 = 1010 nM T63505 C1HSE0 67035086 IC50 = 6400 nM T63505 CWI6K5 67035106 IC50 > 10000 nM T63505 C37NKO 67129970 IC50 = 5330 nM T63505 CK80LJ 67130050 IC50 = 5220 nM T63505 CV63UL 67240318 IC50 > 10000 nM T63505 CWF1M9 68263732 Ki > 15000 nM T63505 C8I7GC 68293638 IC50 > 10000 nM T63505 CD56XK 68293660 IC50 > 10000 nM T63505 C7GRV2 68755406 IC50 = 2750 nM T63505 CAIO65 68796885 IC50 = 51 nM T63505 C5DGR9 69036886 IC50 = 1154 nM T63505 CAOE64 69412987 IC50 = 2877 nM T63505 CH6S7Q 70681377 Ki = 0.7943 nM T63505 C82FIP 70686752 IC50 = 1700 nM T63505 C0QX3Y 70688829 IC50 = 820 nM T63505 CKY12U 70690667 Ki > 10000 nM T63505 CUS3F6 70691280 IC50 > 100000 nM T63505 CSOT12 70693058 IC50 > 10000 nM T63505 CS6NW3 70693059 IC50 > 10000 nM T63505 CL4Z7S 70701950 IC50 = 441 nM T63505 C1IEJ2 70789254 IC50 = 126000 nM T63505 C8T7ZP 70789255 IC50 = 7000 nM T63505 CH0B8N 70789756 IC50 > 30000 nM T63505 C4ML7J 70866004 IC50 = 457 nM T63505 CK2QM6 70866006 IC50 = 165 nM T63505 CJK8F2 70866032 IC50 = 1047 nM T63505 CV74OC 70866036 IC50 = 757 nM T63505 C6MV9L 70866060 IC50 = 3206 nM T63505 CMX75Z 70866164 IC50 = 28 nM T63505 CVNH21 70866177 IC50 = 149 nM T63505 CKJI02 70866181 IC50 = 594 nM T63505 CC98EU 71449991 IC50 = 92.2 nM T63505 CV21PC 71449992 IC50 = 341 nM T63505 CG59TB 71449993 IC50 = 14.2 nM T63505 C23ETA 71450038 IC50 = 12.7 nM T63505 C3B7IP 71450039 IC50 = 0.98 nM T63505 C0XL6Z 71451816 IC50 = 122 nM T63505 CQM05U 71451817 IC50 = 1.12 nM T63505 CVE9P2 71451818 IC50 = 5.09 nM T63505 C30FHU 71453635 IC50 = 25.2 nM T63505 CR7DI8 71453636 IC50 = 89.4 nM T63505 C8K6BL 71453637 IC50 = 486 nM T63505 C12IUO 71453638 IC50 = 2.18 nM T63505 CIEK84 71453639 IC50 = 31.5 nM T63505 C0FTX4 71453675 IC50 = 11.4 nM T63505 CK7V6O 71453676 IC50 = 9.83 nM T63505 CU42QX 71455363 IC50 = 14.4 nM T63505 C4X9GT 71455364 IC50 = 10.6 nM T63505 CVY26H 71455365 IC50 = 29.6 nM T63505 C3X1OP 71455406 IC50 = 18 nM T63505 COUR46 71455407 IC50 = 10.6 nM T63505 C8IV0R 71455408 IC50 = 38.9 nM T63505 CKT60L 71455860 Ki > 700 nM T63505 CY2G7S 71457180 IC50 = 1.94 nM T63505 CXA9W8 71457181 IC50 = 38 nM T63505 CCT0X3 71459003 IC50 = 250 nM T63505 C01XBA 71459004 IC50 = 272 nM T63505 C0WF3X 71459043 IC50 = 7.93 nM T63505 CJ3PO5 71459044 IC50 = 659 nM T63505 CW0X4B 71460798 IC50 = 95.7 nM T63505 CE84WT 71460799 IC50 = 342 nM T63505 CG0F1R 71460800 IC50 = 2130 nM T63505 CZM79U 71460801 IC50 = 206 nM T63505 CWT1E8 71460802 IC50 = 1.22 nM T63505 CZ72YB 71460803 IC50 = 334 nM T63505 C8KL1P 71460845 IC50 = 32.8 nM T63505 C7XZ6K 71460846 IC50 = 130 nM T63505 CS08OH 71462551 IC50 = 0.94 nM T63505 CB45LP 71462552 IC50 = 18.7 nM T63505 CW8JR3 71510528 IC50 = 1530 nM T63505 C9DIK2 71512060 IC50 = 2262 nM T63505 C6HF8S 71521082 IC50 = 2953 nM T63505 C9Z3AI 71521083 IC50 = 749.8 nM T63505 C5ZKU7 71546969 IC50 = 578 nM T63505 C7ARI9 71547113 IC50 = 1282 nM T63505 CCN01X 71547862 IC50 > 10000 nM T63505 C1IT5U 71550931 IC50 = 308 nM T63505 CA3O6K 71552696 IC50 = 910 nM T63505 C1NPL0 71552941 IC50 = 12030 nM T63505 CA4PS8 71552942 IC50 = 16360 nM T63505 C3UA9C 71553011 IC50 = 21110 nM T63505 CEZ15Y 71553012 IC50 = 3170 nM T63505 CVIA91 71553085 IC50 = 7610 nM T63505 C1TR3O 71553152 IC50 = 30000 nM T63505 CDR80A 71562417 IC50 = 1.33 nM T63505 CGQB43 71562418 IC50 = 0.36 nM T63505 CFNY63 71562419 IC50 = 1.28 nM T63505 CDW47A 71562420 IC50 = 2.16 nM T63505 C2P4YC 71562521 IC50 = 0.57 nM T63505 CE3SA8 71562522 IC50 = 0.53 nM T63505 C1NQ0E 71562523 IC50 = 2.07 nM T63505 CQX7B1 71562524 IC50 = 10.58 nM T63505 CC06AT 71562525 IC50 = 2.72 nM T63505 CB6ZT9 71562762 IC50 = 13.9 nM T63505 C24FGW 71562763 IC50 = 0.76 nM T63505 CN7W5S 71579325 IC50 > 10000 nM T63505 C1BCX0 71579696 IC50 = 281 nM T63505 CRC5M0 71605046 IC50 = 1.9 nM T63505 C7GN8S 71605048 IC50 = 0.4 nM T63505 CT90RH 71605222 IC50 = 0.2 nM T63505 CBW27Q 71605223 IC50 = 307 nM T63505 C64OFJ 71605224 IC50 = 30 nM T63505 C4ZHD2 71605225 IC50 = 31 nM T63505 CEL6H2 71605226 IC50 = 22 nM T63505 C3CB5M 71605407 IC50 = 13 nM T63505 C3YL2D 71605408 IC50 = 40 nM T63505 C75QZO 71654679 IC50 = 0.77 nM T63505 CS5V4W 71654755 IC50 = 0.89 nM T63505 CAU6E5 71655122 IC50 = 23.13 nM T63505 C8DTM7 71655275 IC50 = 698.6 nM T63505 CI5TZ1 71655333 IC50 = 139.4 nM T63505 C7T1SU 71655334 IC50 = 953.1 nM T63505 CSVL84 71655335 IC50 = 16.9 nM T63505 C71MBF 71655336 IC50 = 21.4 nM T63505 CA3CV6 71655337 IC50 = 44.9 nM T63505 C4EW2I 71655338 IC50 = 6.2 nM T63505 CA3MN9 71655339 IC50 = 168.2 nM T63505 C1IY5H 71655397 IC50 = 2.3 nM T63505 CU53FZ 71655398 IC50 = 46.7 nM T63505 C6LUD0 71655399 IC50 = 1479 nM T63505 C2CO3B 71655400 IC50 = 45.2 nM T63505 CBH8Z7 71655401 IC50 = 23.2 nM T63505 C7CB3J 71655402 IC50 = 43.1 nM T63505 CIR7W6 71655403 IC50 = 11.2 nM T63505 CM6A1X 71655462 IC50 = 199.6 nM T63505 C15JIZ 71655463 IC50 = 39 nM T63505 CW06NY 71655464 IC50 = 176.6 nM T63505 C21TYX 71655465 IC50 = 171.5 nM T63505 C1NW6B 71655466 IC50 = 239.4 nM T63505 C8Y0DV 71655467 IC50 = 182.5 nM T63505 CYMR36 71655468 IC50 > 100000 nM T63505 C1M4IL 71655525 IC50 > 100000 nM T63505 CE74KM 71655596 IC50 = 6.12 nM T63505 CY9GL5 71655597 IC50 = 0.11 nM T63505 CXW13N 71655598 IC50 = 0.064 nM T63505 C8PFW6 71655599 IC50 = 3.6 nM T63505 C52QNH 71655600 IC50 = 2.8 nM T63505 C74YCW 71655601 IC50 = 15.3 nM T63505 C5PAG6 71655602 IC50 = 14.4 nM T63505 CZ3HR8 71655663 IC50 = 0.31 nM T63505 CPQ03V 71655664 IC50 = 2 nM T63505 CG0OB8 71655665 IC50 = 5.6 nM T63505 CXBN25 71655666 IC50 = 0.11 nM T63505 CQZ48I 71655667 IC50 = 1.2 nM T63505 C3O9WT 71655668 IC50 = 0.51 nM T63505 CR1PX9 71655669 IC50 = 0.021 nM T63505 C80KLG 71655728 IC50 = 0.064 nM T63505 CW9K6Z 71655729 IC50 = 0.16 nM T63505 COIT35 71655730 IC50 = 0.015 nM T63505 C9LX6J 71655731 IC50 = 0.23 nM T63505 CR3GJ8 71655732 IC50 = 0.18 nM T63505 C40QTR 71655733 IC50 = 0.13 nM T63505 C56CBX 71655734 IC50 = 0.12 nM T63505 C7E6YV 71720026 IC50 = 203 nM T63505 CI2D1A 71727972 IC50 = 4310 nM T63505 CUY7B1 71727973 IC50 = 740 nM T63505 CU64JS 71727974 IC50 = 120 nM T63505 C3C4RB 71727975 IC50 = 1230 nM T63505 CZ53TI 71728101 IC50 = 1530 nM T63505 C4UB5Q 71728102 IC50 = 2170 nM T63505 C9KYW6 71728103 IC50 = 1880 nM T63505 CQ4ZR0 71728212 IC50 = 1040 nM T63505 C4EZ7S 71728213 IC50 = 17600 nM T63505 CD3B8G 71728214 IC50 = 820 nM T63505 C3LPX9 71728215 IC50 = 2270 nM T63505 C04KUB 71728216 IC50 = 4310 nM T63505 CI4N7R 71745294 Ki = 1080 nM T63505 CRC14G 71745295 Ki = 2710 nM T63505 CCQE91 71745296 Ki = 99 nM T63505 C5Z8IT 71745297 Ki = 1343 nM T63505 C9D5PT 71745298 Ki = 673 nM T63505 CAJ13X 71745299 Ki = 3400 nM T63505 CN91IU 71745494 Ki = 1155 nM T63505 CE1P4S 71745495 Ki = 60 nM T63505 C9H5ZR 71745496 Ki = 50 nM T63505 C7SUW0 71747648 Ki = 36 nM T63505 CE5KF3 71747828 Ki = 180 nM T63505 C7HJG1 71747829 Ki = 656 nM T63505 CRU82Q 71747830 Ki = 260 nM T63505 CGKP21 71747831 Ki = 1440 nM T63505 CAQ1W4 71747832 Ki = 890 nM T63505 CE3A9T 71747833 Ki = 90 nM T63505 C4GJ1V 71747834 Ki = 575 nM T63505 C14EQL 71748013 Ki = 21 nM T63505 COZT25 71748014 Ki = 2 nM T63505 C6BN2O 71748015 Ki = 29 nM T63505 CHWO28 71748016 Ki = 1500 nM T63505 CUQW27 71748017 Ki = 497 nM T63505 CM82AO 71748018 Ki = 6 nM T63505 CS4E9X 71762922 Ki > 100000 nM T63505 C75QWC 71763641 IC50 = 157 nM T63505 CVJ7S2 71763642 IC50 = 42 nM T63505 C8M4HU 71763643 IC50 = 73 nM T63505 CM4X1R 71763869 IC50 = 1273 nM T63505 CKN96V 71764058 IC50 = 379 nM T63505 C1K5HE 71764059 IC50 = 9 nM T63505 C42VJY 71764060 IC50 = 23 nM T63505 CI9H6L 72164895 Ki = 2350 nM T63505 CB2NP7 72165228 IC50 = 0.5 nM T63505 CD85OH 72201590 IC50 = 11 nM T63505 C5KTR3 72201875 IC50 = 19 nM T63505 C9XL7F 72202747 IC50 = 18 nM T63505 CXLR81 72203284 IC50 = 24 nM T63505 C4E2VS 72543811 IC50 > 50000 nM T63505 C3B0CK 72544445 IC50 = 1.1 nM T63505 C27NJL 72545853 IC50 = 35 nM T63505 C60TUV 72737208 IC50 > 10000 nM T63505 CJ3WA6 72737404 IC50 = 566 nM T63505 C71GBE 73349501 IC50 = 1500 nM T63505 C2PAK9 73438493 IC50 = 20 nM T63505 CHI51J 76070594 IC50 = 170 nM T63505 CB4V1R 76071142 IC50 = 90 nM T63505 CBAT06 76071144 IC50 = 50 nM T63505 C7SH1T 76071506 IC50 = 100 nM T63505 CS87EI 76071624 IC50 = 240 nM T63505 CRK1L2 76210601 IC50 = 250 nM T63505 CH8W7D 77461036 IC50 > 1000 nM T63505 CC4F0A 78319160 IC50 = 15000 nM T63505 CO4IE9 78319161 IC50 = 39000 nM T63505 CY6LN4 78319162 IC50 = 33000 nM T63505 CN7HU3 86288843 IC50 = 5900 nM T63505 C5Y1WO 86288855 IC50 = 5800 nM T63505 CCJ43A 86302281 IC50 > 10000 nM T63505 CB5NJ4 86302541 IC50 > 10000 nM T63505 CPG3A5 86302574 IC50 > 30000 nM T63505 C1HW4B 89735655 IC50 = 9100 nM T63505 C0AK9G 89891791 IC50 = 439 nM T63505 CT7KE8 89891806 IC50 = 37 nM T63505 C73PSN 89891847 IC50 = 30 nM T63505 C6OP5F 89899385 IC50 = 805 nM T63505 CBW32H 89899386 IC50 = 131 nM T63505 C9W7ZN 89899405 IC50 = 136 nM T63505 CTY2A0 89899410 IC50 = 3000 nM T63505 CPVZ54 89899415 IC50 = 5.3 nM T63505 CJYP54 89899416 IC50 = 515 nM T63505 CSM02W 89899417 IC50 = 1.4 nM T63505 CDAU89 89899421 IC50 = 19 nM T63505 C5RAI0 89907349 IC50 = 4 nM T63505 CP0GY3 89908140 IC50 < 0.3 nM T63505 C0JA2V 89908303 IC50 = 0.4 nM T63505 CJW7L6 89908440 IC50 = 1.6 nM T63505 CFB75T 90479825 IC50 = 206 nM T63505 CY0UC4 90645194 IC50 > 10000 nM T63505 C3GU7P 90645237 IC50 > 10000 nM T63505 CFI93O 90645239 IC50 > 10000 nM T63505 C76KSB 90645241 IC50 > 10000 nM T63505 CNWP80 90645243 IC50 > 10000 nM T63505 C1POJ2 90645244 IC50 > 10000 nM T63505 C8BEX4 90645245 IC50 > 10000 nM T63505 CW0L1D 90654798 IC50 > 25000 nM T63505 CDF2A1 90654799 IC50 > 50000 nM T63505 CO2CU1 90654800 IC50 = 20000 nM T63505 C4NXO7 90654801 IC50 = 34000 nM T63505 CE54MK 90654802 IC50 > 50000 nM T63505 C5PO6N 90654803 IC50 > 25000 nM T63505 CID9U2 90654804 IC50 > 50000 nM T63505 CX29IY 90655145 IC50 > 10000 nM T63505 CU31VY 90675933 IC50 > 50000 nM T63505 C2XWG7 90675934 IC50 > 50000 nM T63505 CH7R2B 90675935 IC50 > 50000 nM T63505 CORQ94 90675936 IC50 > 25000 nM T63505 CE39DC 90675937 IC50 > 50000 nM T63505 CSU5K2 90675938 IC50 = 5900 nM T63505 CE8S1J 90675939 IC50 > 50000 nM T63505 C1H9FB 90675940 IC50 > 50000 nM T63505 CPB36R 90675941 IC50 > 50000 nM T63505 C41DFX 101913643 Ki = 120 nM T63505 CQ9PN8 102593934 IC50 = 8700 nM T63505 CAI09J 118195093 IC50 = 0.5 nM T63505 CZ5G7W 118195200 IC50 = 2.3 nM T63505 C0NM1V 118195331 IC50 = 18 nM T63505 C3J4UQ 118198923 IC50 = 7 nM T63505 C9MJE1 118226293 Ki = 0.103 nM T63505 CP40JF 118722001 IC50 > 50000 nM T63505 C4DU6M 118725835 Ki = 130 nM T63505 CA9GJ0 118725874 Ki = 430 nM T63505 CJST86 118725875 Ki = 150 nM T63505 C25DKS 118725880 Ki = 120 nM T63505 CO4CN9 118725884 Ki = 150 nM T63505 CI7MY8 118728501 IC50 > 100000 nM T63505 CZE9K8 118728502 IC50 > 100000 nM T63505 C6F5PQ 119081684 IC50 > 10000 nM T63505 CKBP72 121231408 IC50 = 479 nM T63505 CN4X0C 121231414 IC50 > 10000 nM T63505 C1Y7UH 121305843 Ki > 100000 nM T63505 CHG8Y6 121316022 Ki > 100000 nM T63505 C81IFQ 122163152 IC50 > 100000 nM T63505 C08KEM 122179540 IC50 = 3800 nM T63505 CG0RP7 122179547 IC50 = 2400 nM T63505 C1A0SQ 122179548 IC50 = 5200 nM T63505 CCXA46 122190499 Ki = 980 nM T63505 C3PQ4W 122190505 Ki = 730 nM T63505 CN1DK0 122190507 Ki = 1200 nM T63505 C4X7SD 122192466 IC50 > 10000 nM T63505 CN41IF 122634050 IC50 = 70 nM T63505 CD67LU 122705248 IC50 = 116 nM T63505 CX63VW 122705258 IC50 = 7249 nM T63505 C76IKM 122705261 IC50 = 1207 nM T63505 CY30FL 123752658 IC50 = 23.2 nM T63505 C8ALO2 124088839 IC50 = 7525 nM T63505 CK46IZ 124088840 IC50 = 10000 nM T63505 CKC81N 124088842 IC50 = 9440 nM T63505 C2XIS6 124088843 IC50 > 10000 nM T63505 CXVU91 124088862 IC50 > 10000 nM T63505 COBA69 124088864 IC50 = 370 nM T63505 CBLA08 124088870 IC50 = 808 nM T63505 CX3O4K 124088871 IC50 > 10000 nM T63505 C4OH5B 124088876 IC50 = 2950 nM T63505 C8KXV1 127025843 IC50 > 1000 nM T63505 C0HN2Y 127030123 IC50 = 25150 nM T63505 C7S9GI 127030124 IC50 > 100000 nM T63505 CHGN68 127030424 IC50 = 2540 nM T63505 CRV62L 127030425 IC50 = 22520 nM T63505 CF7JT8 127030426 IC50 = 7910 nM T63505 C5YCU2 127030427 IC50 > 100000 nM T63505 C0GES2 127031075 IC50 = 30830 nM T63505 CFJ32Y 127031076 IC50 > 100000 nM T63505 CC8V4J 127031368 IC50 = 12900 nM T63505 C78GYH 127031383 IC50 = 16610 nM T63505 C5WA9Z 127031384 IC50 > 100000 nM T63505 CD7LN1 127031385 IC50 = 2660 nM T63505 CI0VX4 127031386 IC50 = 11520 nM T63505 CO89TC 127031387 IC50 = 1340 nM T63505 CAM4S5 127031675 IC50 = 5370 nM T63505 C4QD0M 127031676 IC50 = 8710 nM T63505 C0LTC3 127031677 IC50 > 100000 nM T63505 CO1G2K 127032542 IC50 > 100000 nM T63505 C12IOL 127033165 IC50 > 100000 nM T63505 C5RO0L 127033758 IC50 > 100000 nM T63505 CD04YX 127034308 IC50 > 100000 nM T63505 C6KM3T 127034964 IC50 = 0.6 nM T63505 C1BZ4L 127034965 IC50 = 1.1 nM T63505 CBM8A3 127035575 IC50 = 1430 nM T63505 C7O8LT 127035889 IC50 = 1900 nM T63505 CD0P9K 127036142 IC50 = 900 nM T63505 C1C7BZ 127036143 IC50 > 100000 nM T63505 CNKI42 127036144 IC50 = 2700 nM T63505 CYT9O5 127036145 IC50 = 970 nM T63505 CBC35P 127036146 IC50 = 20 nM T63505 C31DNU 127036327 IC50 = 570 nM T63505 C9JZS1 127036328 IC50 = 3 nM T63505 C3IE4T 127036881 IC50 = 270 nM T63505 CKX40V 127037812 IC50 > 10000 nM T63505 C70RUP 127038480 IC50 > 10000 nM T63505 C3WCN8 127041777 IC50 > 10000 nM T63505 C4YF8R 127043007 IC50 > 25000 nM T63505 CSZ13Q 127043201 IC50 > 100000 nM T63505 C9A6RW 127043202 IC50 > 100000 nM T63505 CS3W8L 127043203 IC50 > 12500 nM T63505 C1M3DA 127043204 IC50 > 25000 nM T63505 C2Q4GC 127043205 IC50 > 100000 nM T63505 C2C7OH 127043366 IC50 > 50000 nM T63505 C67EYU 127043440 IC50 > 50000 nM T63505 C36PAN 127043441 IC50 > 50000 nM T63505 C5U7NS 127043619 IC50 > 100000 nM T63505 CYPW41 127043620 IC50 > 25000 nM T63505 C24AYP 127043621 IC50 > 50000 nM T63505 CH82XJ 127043781 IC50 > 12500 nM T63505 CSJ9Z4 127043911 IC50 > 12500 nM T63505 C3JVC4 127044692 IC50 > 50000 nM T63505 CK6E2I 127045497 IC50 > 50000 nM T63505 CG8DA9 127045861 IC50 = 9920 nM T63505 CHK16Q 127045929 IC50 > 1000 nM T63505 CC4ND8 127046862 IC50 = 8630 nM T63505 CY3J0C 127047591 IC50 > 1000 nM T63505 COPL97 127049453 IC50 = 407 nM T63505 CDP32G 127050839 IC50 = 4690 nM T63505 CGT0B1 127052321 IC50 > 10000 nM T63505 CO25WH 127052538 IC50 = 6323 nM T63505 CF5D2Y 129318936 IC50 > 10000 nM T63505 C2LWZ1 129318964 IC50 > 10000 nM T63505 CI9H2W 130364450 IC50 > 10000 nM T63505 C28CLN 130364457 IC50 > 10000 nM T63505 CO9C5Q 130364468 IC50 > 10000 nM T63505 CBI35E 132275094 IC50 = 3 nM T63505 C6ROQ3 132546210 IC50 = 46 nM T63505 CERS64 132937256 IC50 > 30000 nM T63505 CHLJ63 134132321 IC50 = 150000 nM T63505 C98MZB 134132731 IC50 = 20900 nM T63505 CZG2L5 134135232 IC50 = 12200 nM T63505 CB3SZ2 134135265 IC50 = 7252 nM T63505 C32AGN 134136205 IC50 = 7 nM T63505 CM68VX 134143486 IC50 = 40000 nM T63505 C7SL4N 134143939 IC50 = 19000 nM T63505 CN35SO 134146628 IC50 > 1000 nM T63505 C06SFD 134150115 IC50 = 65600 nM T63505 CR4QC3 134152617 IC50 = 30 nM T63505 CGDL39 134155715 IC50 = 6 nM T63505 C2YJ7D 134156776 IC50 = 110000 nM T63505 C6NFD0 134419123 IC50 = 2000 nM T63505 C1X6FJ 134693894 IC50 = 494 nM T63505 CYL5V1 134694986 IC50 > 30000 nM T63505 C3K5PA 134814272 IC50 = 550 nM T63505 CLCO61 135398510 IC50 = 450 nM T63505 CVJK60 135402835 IC50 = 240 nM T63505 C5BPY7 135402910 IC50 > 500000 nM T63505 CU60YC 135431661 IC50 = 1100 nM T63505 C46QAS 135441185 IC50 = 10 nM T63505 C19YWA 135457035 Ki = 520 nM T63505 C08KLE 135520206 Ki = 5 nM T63505 CZFA70 135611366 IC50 = 478 nM T63505 CU29YK 135750268 IC50 = 1700 nM T63505 C0PVG7 135819982 IC50 = 30 nM T63505 C9ZI5J 135820026 IC50 = 30 nM T63505 C2PJK6 135820173 IC50 = 7 nM T63505 C53LFX 135820297 IC50 = 60 nM T63505 CBLH60 135820360 IC50 = 230 nM T63505 C5BI9T 135820431 IC50 = 200 nM T63505 CP7KZ8 135820466 IC50 = 130 nM T63505 CQK62L 135820498 IC50 = 150 nM T63505 C4PD2G 135820511 IC50 = 60 nM T63505 CJV08H 135897884 IC50 = 4564 nM T63505 C4K3XL 135897887 IC50 = 7.2 nM T63505 C93QJC 135897888 IC50 = 34.1 nM T63505 CX6JV7 135897894 IC50 = 66.9 nM T63505 C5QUL0 135897897 IC50 = 0.87 nM T63505 CLV7Y8 135897900 IC50 = 10.2 nM T63505 CFJZ14 135897904 IC50 = 3440 nM T63505 CT2UV5 135897905 IC50 = 468 nM T63505 C12UDA 135947972 IC50 = 664 nM T63505 CN42ZS 135947973 IC50 = 70 nM T63505 CF8AO3 135947974 IC50 = 1900 nM T63505 CW08GJ 135947976 IC50 = 328 nM T63505 CJN7E2 135947978 IC50 = 1500 nM T63505 CFKH34 135947979 IC50 = 57 nM T63505 C0G1UL 135998453 Ki = 280 nM T63505 C5XIE8 136026041 IC50 = 7800 nM T63505 C4E2DO 136038437 IC50 = 900 nM T63505 CL3KN6 136038471 IC50 = 20 nM T63505 CQ9TJ0 136038505 IC50 = 220 nM T63505 CL5H2C 136038513 IC50 = 60 nM T63505 CVI17Q 136038596 IC50 = 3 nM T63505 CAXJ50 136043793 IC50 = 600 nM T63505 CAW0E4 136065882 IC50 > 100000 nM T63505 CVIC49 136069671 IC50 = 1500 nM T63505 CZ7EX0 136183413 IC50 = 7680 nM T63505 C5X7SM 137228145 IC50 > 50000 nM T63505 CUF6V2 137228146 IC50 > 50000 nM T63505 CJGO41 137228147 IC50 > 25000 nM T63505 C4W6IF 137228148 IC50 > 25000 nM T63505 CA27JH 137228149 IC50 > 25000 nM T63505 CH0T8X 137228150 IC50 > 100000 nM T63505 CY3HX8 137228151 IC50 > 50000 nM T63505 CTRM24 137228152 IC50 > 50000 nM T63505 CUK42G 137228153 IC50 > 50000 nM T63505 C5M0WE 137228154 IC50 > 50000 nM T63505 CXC69T 137321158 IC50 = 335 nM T63505 C25ERN 137631967 IC50 = 4.3 nM T63505 CI1E8V 137634241 IC50 = 408 nM T63505 C79XWZ 137636138 Ki > 100000 nM T63505 C8GQD5 137636872 IC50 = 20 nM T63505 C06JRX 137637094 IC50 = 2.9 nM T63505 C7KQH8 137644946 IC50 = 70000 nM T63505 C1DK0P 137651391 IC50 = 6.1 nM T63505 C28QUP 137652864 IC50 = 801.5 nM T63505 CV5H3Z 137657932 IC50 = 6.6 nM T63505 CS61AX 137659496 IC50 > 100000 nM T63505 CM3UF7 137700779 IC50 > 10000 nM T63505 C3K5LU 137796291 IC50 > 10000 nM T63505 C0B8GK 138377594 IC50 = 360 nM T63505 C2JI6T 138393294 IC50 = 156 nM T63505 C0PYR1 138454771 IC50 = 2 nM T63505 CN0X5D 138454787 IC50 = 1340 nM T63505 CSRI06 138547901 IC50 > 1000 nM T63505 CUXO19 138617501 IC50 > 1000 nM T63505 CMA0E6 138753300 IC50 = 398.11 nM T63505 C6VB3O 145925651 IC50 >= 5000 nM T63505 C29XUO 145945978 IC50 > 1000 nM T63505 C7SH9V 145949579 IC50 = 9.4 nM T63505 CQCV54 145950906 IC50 = 7700 nM T63505 CKWZ34 145950923 IC50 = 21.1 nM T63505 CGOE73 145951398 IC50 = 564 nM T63505 CZF70O 145951916 IC50 = 30.2 nM T63505 CNK12Z 145952731 IC50 = 932 nM T63505 CGV16H 145954003 IC50 > 10000 nM T63505 CG46IU 145954838 IC50 = 340 nM T63505 CUIT87 145955254 IC50 = 97.4 nM T63505 CX2U6N 145956375 IC50 = 346 nM T63505 CC0RU9 145956925 IC50 = 9700 nM T63505 CA2F0O 145958559 IC50 = 11.94 nM T63505 C12VOP 145959821 IC50 > 10000 nM T63505 C5PZ9J 145959874 IC50 = 281 nM T63505 CF0C6K 145960274 IC50 = 21 nM T63505 C8NDS6 145971939 IC50 = 202 nM T63505 CP9NB6 145974090 IC50 > 10000 nM T63505 CBR08X 145983359 IC50 = 3.5 nM T63505 CE2X6V 145983518 IC50 = 10 nM T63505 C4ID8J 145984666 IC50 = 7 nM T63505 CW6ZJ2 145984860 IC50 = 22 nM T63505 CI85EU 145998085 IC50 = 1369 nM T63505 C05WAM 146344085 IC50 > 1000 nM T63505 CV2DX0 152875297 IC50 = 794.33 nM T63505 C5MP1Q 155510890 IC50 > 10000 nM T63505 C0TUR6 155511823 IC50 = 251.19 nM T63505 CA10CQ 155512867 IC50 > 1000 nM T63505 C2MD1Q 155513187 IC50 > 10000 nM T63505 C5B2AX 155513312 IC50 > 1000 nM T63505 CM9V5R 155513533 Ki = 0.49 nM T63505 CZMD64 155514443 IC50 > 1000 nM T63505 CRGM52 155515395 IC50 = 251.19 nM T63505 CPFY91 155516930 IC50 = 1995.26 nM T63505 C1JNF5 155516932 IC50 = 251.19 nM T63505 CEL62J 155517148 IC50 = 39.81 nM T63505 CWL3E1 155518230 EC50 = 100 nM T63505 CIU1T6 155518465 IC50 > 1000 nM T63505 C86HPW 155518524 IC50 = 69000 nM T63505 C18WRZ 155519259 IC50 = 25118.86 nM T63505 CQ1PY6 155519503 IC50 = 125.89 nM T63505 CO63MP 155519543 IC50 > 1000 nM T63505 CDN2K5 155519550 IC50 = 1584.89 nM T63505 C5R2WC 155521519 IC50 = 398.11 nM T63505 C9BM4L 155521549 IC50 = 794.33 nM T63505 CHX98P 155522217 Ki = 0.507 nM T63505 CBG4P0 155524103 IC50 > 1000 nM T63505 CBEA43 155524177 IC50 = 31.62 nM T63505 C81VBU 155524466 IC50 = 251.19 nM T63505 C8YLF0 155525255 IC50 = 15848.93 nM T63505 C34XCT 155525282 IC50 = 3162.28 nM T63505 CDI0E3 155527028 IC50 = 2511.89 nM T63505 C3P8QE 155527943 Ki = 0.35 nM T63505 CN6C2T 155528463 IC50 > 1000 nM T63505 C0HW7F 155530527 IC50 > 1000 nM T63505 CP5IW9 155530600 IC50 > 1000 nM T63505 C90DEG 155531134 IC50 = 398.11 nM T63505 CG4BX3 155532203 IC50 = 398.11 nM T63505 C3MC2P 155532434 IC50 = 449.1 nM T63505 CNE6A3 155532801 IC50 > 1000 nM T63505 C2KAU0 155533663 IC50 > 1000 nM T63505 C16YZS 155534423 Ki = 0.418 nM T63505 CV9D5J 155536164 IC50 > 1000 nM T63505 C3LC9I 155536820 IC50 = 930.8 nM T63505 C3X2ZR 155537965 EC50 = 1584.89 nM T63505 C3V4LG 155538413 IC50 = 182 nM T63505 CPG5T4 155538560 IC50 > 10000 nM T63505 C08CGK 155541742 IC50 = 0.2 nM T63505 C5F8EP 155542472 IC50 = 1995.26 nM T63505 CJKS54 155543738 IC50 = 1584.89 nM T63505 CZB7W2 155545289 IC50 = 125.89 nM T63505 CRV40J 155546026 IC50 > 1000 nM T63505 CDIV25 155547658 IC50 = 794.33 nM T63505 CZ56YB 155548149 IC50 > 100000 nM T63505 CCJ9F4 155548184 IC50 = 199.53 nM T63505 CJ6B8R 155548768 IC50 = 630.96 nM T63505 CULE86 155548799 IC50 = 158.49 nM T63505 CSPY71 155548988 IC50 = 158.49 nM T63505 C31WML 155548991 IC50 = 1584.89 nM T63505 C8AG4U 155550655 IC50 > 1000 nM T63505 C14QWH 155551649 IC50 > 10000 nM T63505 C52XGB 155552833 IC50 = 125.89 nM T63505 C8O1QC 155558112 IC50 = 125.89 nM T63505 C7N1AT 155560186 IC50 > 10000 nM T63505 C7E9TC 155560199 IC50 = 1000 nM T63505 CBV70S 155560614 IC50 = 251.19 nM T63505 CU3YH6 155561237 IC50 = 1000 nM T63505 C2QC5F 155562643 IC50 > 10000 nM T63505 CWR4O5 155565233 IC50 > 1000 nM T63505 CRFW02 155566430 IC50 = 33.31 nM T63505 CW3A9B 155566800 EC50 = 501.19 nM T63505 CRPH84 155568071 IC50 = 2511.89 nM T63505 D00ATA 5908088 IC50 > 50000 nM T63505 D00ERW 44444843 Ki > 706 nM T63505 D00HVA 11624601 Ki > 710 nM T63505 D00TBD 10461815 IC50 = 1400 nM T63505 D00TVY 44300176 IC50 = 1800 nM T63505 D01GNF 10301426 Ki = 800 nM T63505 D02BXJ 46864270 IC50 = 0.2 nM T63505 D03DZO 11715767 IC50 > 10000 nM T63505 D03EHM 24905142 IC50 = 2 nM T63505 D03GQI 1049055 Ki = 600 nM T63505 D03NPX 447077 Ki = 0.2 nM T63505 D04QUI 2250919 Ki = 2500 nM T63505 D05FXD 44478401 IC50 = 0.92 nM T63505 D05UJT 5311510 IC50 = 9 nM T63505 D06CYG 44300143 IC50 = 2900 nM T63505 D06HVH 54613583 IC50 > 10000 nM T63505 D07ADX 54764565 IC50 = 3 nM T63505 D07LYJ 1075248 Ki = 1000 nM T63505 D07OSK 6419834 IC50 = 19000 nM T63505 D08HFG 24809764 IC50 > 10000 nM T63505 D09QKH 1097674 Ki = 1300 nM T63505 D0A5MG 1094114 Ki = 2000 nM T63505 D0CE3R 5312137 IC50 > 50000 nM T63505 D0D3RL 44517649 IC50 = 400 nM T63505 D0D8OY 25210550 IC50 = 20 nM T63505 D0D8ZN 1728080 Ki = 5000 nM T63505 D0E7VO 59627005 IC50 = 1.2 nM T63505 D0EE6A 6398883 IC50 = 2820 nM T63505 D0GT8N 5154691 IC50 = 120 nM T63505 D0GW4Q 5330524 IC50 = 21 nM T63505 D0H1OK 11562302 Ki = 19.4 nM T63505 D0H2CM 135565635 IC50 = 410 nM T63505 D0H3RD 44412060 Ki = 400 nM T63505 D0I3XZ 11601743 IC50 = 1300 nM T63505 D0JR3W 71605047 IC50 = 0.2 nM T63505 D0M9QM 5327820 IC50 > 10000 nM T63505 D0O6OH 71553154 IC50 = 810 nM T63505 D0P3JW 447700 IC50 = 2.8 nM T63505 D0Q3NG 11715520 Ki > 710 nM T63505 D0R2WK 16038120 IC50 = 1048 nM T63505 D0S7IE 11658882 Ki > 710 nM T63505 D0T8NU 16757525 IC50 > 4000 nM T63505 D0UN9O 3385203 IC50 >= 10000 nM T63505 D0US9O 45275255 IC50 = 25 nM T63505 D0W7TU 947057 IC50 > 50000 nM T63505 D0Y1UL 10561847 IC50 > 50000 nM T63505 D0YZ7H 9797370 IC50 = 22 nM T65236 D08QMX 5757 EC50 = 0.3 nM T65236 CE6D5B 25481402 EC50 = 20 nM T65236 CZ76MC 71937602 EC50 = 1620 nM T65236 C1W6EX 135351819 EC50 = 480 nM T65236 D02WIL 7433743 IC50 = 20 nM T65236 D0WM5O 5322399 EC50 = 2 nM T24965 D0OB1J 39186 Ki = 380 nM T24965 C7GZ4C 9885728 Ki = 540 nM T24965 CPR12J 10252898 Ki = 42 nM T24965 C07PWG 15612145 Ki = 650 nM T24965 CL2NQ9 44327284 Ki = 85 nM T70036 D0Y6UB 10130754 Ki = 1.4 nM T70036 C2MG9X 9797132 Ki = 8 nM T70036 C0S8LP 11152839 Ki = 14.9 nM T70036 CK39MU 11221621 Ki = 0.9 nM T70036 C0L9YE 11244530 Ki = 14.4 nM T70036 C98AHT 11244637 Ki = 12 nM T70036 C0ER6M 11258369 Ki = 95.3 nM T70036 C5X7AU 11325495 Ki = 939 nM T70036 C14FPS 11393150 Ki = 2.1 nM T70036 C3AS4T 11395389 Ki = 2711 nM T70036 CG2P6K 11405975 Ki = 4388 nM T70036 C4TEO7 11416756 Ki = 1109 nM T70036 CX1U5E 11429402 Ki = 5.3 nM T70036 CZ4JC3 11439226 Ki = 5.9 nM T70036 C6RUL8 11484828 Ki = 1285 nM T70036 C4AW5G 11751841 Ki > 100000 nM T70036 CEY2J1 11784768 Ki = 4434 nM T70036 CI8UA2 44293359 Ki = 392 nM T70036 CX6NB7 118718108 Ki = 335 nM T70036 D06JOJ 10043679 Ki = 3 nM T40276 D01XYJ 35370 IC50 > 150000 nM T40276 D06IAR 60961 IC50 = 278000 nM T40276 D02RJY 11442891 IC50 > 10000 nM T40276 D03HUX 49792852 IC50 > 10000 nM T40276 D09DHT 27924 Ki = 1.8 nM T40276 D0E3TC 44259 IC50 = 1.44 nM T40276 D0I6VU 176167 IC50 = 6 nM T40276 D0LF1U 5287969 IC50 > 45000 nM T40276 D0MS3Z 16725726 IC50 = 19 nM T40276 D0O0LS 25141092 IC50 > 1000 nM T40276 D0Q9UX 16718576 IC50 > 10000 nM T40276 D0R9YR 64971 IC50 > 150000 nM T40276 D0S5RC 3025986 IC50 > 40000 nM T40276 D0W3LI 153999 IC50 = 4.7 nM T40276 D0Z1DH 10029385 IC50 = 420 nM T40276 D03BNU 59604787 IC50 > 10000 nM T40276 D0WS1V 448991 IC50 > 100000 nM T40276 D04FHB 6918852 Ki > 5000 nM T40276 D0A9KI 9863367 IC50 = 17 nM T40276 D0R2TM 5287736 IC50 = 10 nM T40276 D0T3ME 156422 IC50 = 6900 nM T40276 D0X0HN 15391529 IC50 = 270 nM T40276 C8OI7N 2290 IC50 = 10 nM T40276 C91OFE 64980 IC50 > 150000 nM T40276 CG2P1X 159320 Ki = 0.4 nM T40276 C8PU1O 188534 Ki = 9.8 nM T40276 C1ZG2U 449087 IC50 > 10000 nM T40276 C6DLK3 644364 IC50 = 2800 nM T40276 CTID76 5282335 IC50 > 45000 nM T40276 CLA43B 5327919 IC50 = 220 nM T40276 CPDC54 5327920 IC50 = 2200 nM T40276 CCB9G3 5327921 IC50 = 10 nM T40276 CRTQ98 5327922 IC50 = 40 nM T40276 CP20NQ 5327923 IC50 = 6900 nM T40276 C98CNM 5327943 IC50 = 4500 nM T40276 C61URB 5327944 IC50 = 40 nM T40276 CWUY53 5327945 IC50 = 70 nM T40276 CQ54BE 5327946 IC50 = 220 nM T40276 CIB3P0 5327947 IC50 = 20 nM T40276 CVG0A1 5327948 IC50 = 30 nM T40276 C8M3PD 5327949 IC50 = 220 nM T40276 CA25BM 5327950 IC50 = 2800 nM T40276 COP0Q2 5327951 IC50 = 500 nM T40276 CB47VN 5327952 IC50 = 210 nM T40276 CPO51K 5327953 IC50 = 40 nM T40276 CI6AY9 5327954 IC50 = 3600 nM T40276 C1Q0PM 5327955 IC50 = 2800 nM T40276 CXA23M 5327956 IC50 = 830 nM T40276 CH73DT 5327957 IC50 = 960 nM T40276 CTI6K8 5327963 IC50 = 750 nM T40276 CAO1N9 5327979 IC50 = 290 nM T40276 CMP3X8 5327994 IC50 = 50 nM T40276 C4DG8Y 5327995 IC50 = 150 nM T40276 CDL0S2 5327996 IC50 = 46000 nM T40276 CC43JH 5327997 IC50 = 4800 nM T40276 CKS8M6 5327998 IC50 = 290 nM T40276 CQ7OZ6 5327999 IC50 = 1300 nM T40276 CQWO93 5328000 IC50 = 3500 nM T40276 CU73IX 5328002 IC50 = 290 nM T40276 CTVP40 5328003 IC50 = 1000 nM T40276 CBSP34 5328004 IC50 = 2200 nM T40276 CS78OD 5328005 IC50 = 20000 nM T40276 CO9YQ6 5328006 IC50 = 22000 nM T40276 CVX2L3 5328007 IC50 = 20 nM T40276 CPD1U9 5328008 IC50 = 20 nM T40276 C3X6QJ 5328012 IC50 = 1600 nM T40276 CZO4E1 5328013 IC50 = 440 nM T40276 CZ3LK2 5330387 IC50 > 10000 nM T40276 CRU94N 5330388 IC50 > 10000 nM T40276 CDB68F 5330389 IC50 > 10000 nM T40276 CF01JS 5330804 IC50 > 100000 nM T40276 C2RA4O 5352033 Ki = 0.17 nM T40276 CBT0X5 9797847 IC50 = 9000 nM T40276 C4PA5X 9800852 Ki = 701 nM T40276 C8J1OL 9826373 IC50 = 30 nM T40276 CP17TY 9847089 IC50 = 3 nM T40276 C0VM9W 9854502 IC50 ~ 100000 nM T40276 CCJK12 9865633 Ki = 17.4 nM T40276 C20NKA 9889351 IC50 = 10 nM T40276 CQD2W7 9935079 IC50 = 6 nM T40276 CK27DN 9948862 IC50 = 939 nM T40276 CP5NJ3 9952970 Ki = 58.2 nM T40276 CV34AB 9958125 IC50 = 30 nM T40276 CJ84TX 9977154 IC50 = 730 nM T40276 C2W3AV 9995236 IC50 = 1500 nM T40276 CJ2EP9 9999648 IC50 = 4360 nM T40276 C5XU8E 10000872 IC50 = 270 nM T40276 C57DLH 10001523 IC50 = 1160 nM T40276 C84CYF 10001880 IC50 = 1850 nM T40276 CBT2P7 10001889 IC50 = 1070 nM T40276 CV7Z9Y 10002471 IC50 = 240 nM T40276 CUY0F8 10005715 IC50 > 10000 nM T40276 CY65CO 10030073 IC50 = 330 nM T40276 C2UGV9 10030483 IC50 = 2500 nM T40276 CO5KL3 10072710 IC50 = 890 nM T40276 CINF40 10073694 IC50 = 2260 nM T40276 CF1D6Y 10075240 IC50 > 10000 nM T40276 CT6BJ7 10099352 IC50 > 150000 nM T40276 CG7JO8 10099482 IC50 = 3800 nM T40276 C93LPQ 10099652 IC50 = 26 nM T40276 CEF8U5 10117705 IC50 = 41 nM T40276 CRT67V 10119173 IC50 = 40 nM T40276 C2O7ZH 10137972 IC50 = 2 nM T40276 CZJI60 10141037 IC50 = 1163 nM T40276 C94WRY 10143231 IC50 > 10000 nM T40276 C76TVG 10143584 IC50 = 29 nM T40276 CLBD08 10144909 IC50 = 18 nM T40276 C7JP1A 10163439 IC50 = 7 nM T40276 C3QZV8 10184859 IC50 = 46 nM T40276 CJN72C 10185160 IC50 = 10 nM T40276 CJ0R2G 10187378 IC50 = 37 nM T40276 C73LXY 10188021 IC50 = 170 nM T40276 CK7UT9 10188786 IC50 = 92 nM T40276 C5P8JC 10206423 IC50 = 46 nM T40276 CGOT91 10207821 IC50 = 9 nM T40276 CUF0W9 10207822 IC50 = 45 nM T40276 C98TUI 10208507 IC50 = 17 nM T40276 C51SKM 10209082 IC50 = 5 nM T40276 CK72XG 10209108 IC50 = 92 nM T40276 C3VK7T 10229967 IC50 = 27 nM T40276 C9HJ3N 10248940 IC50 = 1100 nM T40276 CC7P0T 10272623 IC50 = 220 nM T40276 C7SFI1 10296883 IC50 = 2 nM T40276 CTXN56 10296960 IC50 = 23 nM T40276 CMK32F 10300534 IC50 > 150000 nM T40276 CAX9W2 10302405 IC50 = 7 nM T40276 CNE1H0 10318765 IC50 = 2380 nM T40276 C3IJR7 10339551 IC50 = 1440 nM T40276 CHB84X 10341165 IC50 = 2730 nM T40276 CFU38G 10363814 Ki = 2070 nM T40276 CEH41V 10392789 IC50 = 4 nM T40276 C3RBY8 10395226 Ki = 13.4 nM T40276 CRVE78 10411641 IC50 = 1880 nM T40276 CDR7X8 10415328 IC50 > 150000 nM T40276 CQXJ51 10425978 Ki = 179.5 nM T40276 C36QRS 10453829 Ki = 539 nM T40276 C10PAC 10460251 IC50 = 3 nM T40276 C25LDK 10460643 IC50 = 39000 nM T40276 C1VI3E 10477747 IC50 = 47 nM T40276 CMA4J8 10479260 Ki = 1052 nM T40276 C70SUP 10482065 IC50 > 150000 nM T40276 CX7S8N 10482293 IC50 = 2 nM T40276 C76QGP 10506540 IC50 = 20 nM T40276 CSR8Y5 10527068 IC50 = 48 nM T40276 CDNP37 10530708 IC50 = 20 nM T40276 C5EYJ3 10554684 IC50 = 880 nM T40276 C71UIS 10555532 IC50 = 3600 nM T40276 CZ8UA9 10650891 IC50 = 44 nM T40276 CJOU71 10671412 IC50 = 5 nM T40276 CM5B6A 10673286 IC50 = 38 nM T40276 CN9I6T 10768377 IC50 = 24 nM T40276 CL8VH3 10768554 IC50 = 330 nM T40276 C5YMK8 10769011 IC50 = 5 nM T40276 C7HPA0 10864309 IC50 = 200 nM T40276 C1DRE5 10884145 IC50 = 49 ug.mL-1 T40276 C2G5CU 10894726 Ki > 10000 nM T40276 C1L4ZC 10940039 IC50 = 24 nM T40276 CR47CD 11025838 Ki = 610 nM T40276 C67CSJ 11201611 IC50 = 6.8 nM T40276 C3ROM0 11247414 IC50 = 0.7 nM T40276 C30PKR 11248978 IC50 = 1100 nM T40276 CNBX16 11270660 IC50 > 10000 nM T40276 CSXY78 11294864 IC50 = 560 nM T40276 CRZ38O 11315034 IC50 = 133 nM T40276 CPU9I3 11316975 IC50 = 1000 nM T40276 CQ8I4H 11328863 IC50 = 800 nM T40276 C4ON7Z 11362429 IC50 = 3.4 nM T40276 C8DNQ2 11453012 IC50 = 30 nM T40276 C3KAC4 11538477 IC50 = 42 nM T40276 C1CD2N 11547825 IC50 = 15 nM T40276 C9OV5S 11561609 IC50 = 2.9 nM T40276 CACS26 11561968 Ki > 2000 nM T40276 CD7PF5 11574473 IC50 = 43 nM T40276 CA9XJ2 11604381 IC50 = 1.4 nM T40276 C91XGQ 11612470 IC50 = 1.4 nM T40276 CI9HQ2 11624816 IC50 = 75 nM T40276 CQ5S3G 11639520 IC50 = 93 nM T40276 CP04JC 11666231 IC50 > 10000 nM T40276 CU0E8O 11690457 Ki > 2000 nM T40276 CB0AP2 11705863 Ki > 10000 nM T40276 CCX53Q 11729563 IC50 = 10 nM T40276 CP7AH3 11755812 IC50 = 50000 nM T40276 C17SIL 11756581 IC50 > 150000 nM T40276 CM10YB 11799388 IC50 = 44 nM T40276 C9JT4S 11847343 IC50 = 1212 nM T40276 CTN96I 11851810 IC50 = 0.6 nM T40276 CA05OS 11972484 IC50 = 80 nM T40276 CQ39BY 12115602 IC50 = 2.1 nM T40276 C2BX8F 15297223 IC50 = 30 nM T40276 CE04YW 15297224 IC50 = 4900 nM T40276 C9TU1O 16046126 IC50 > 1000 nM T40276 CC24KI 16667248 IC50 = 27 nM T40276 C6NV2U 17814686 IC50 = 2448 nM T40276 CFAR38 17814740 IC50 = 18 nM T40276 C9AVK0 21113469 IC50 = 60 nM T40276 CS15LY 21672114 Ki = 0.45 nM T40276 CZ0X8J 22592015 IC50 > 315 nM T40276 CVR9K4 22907281 IC50 = 19 nM T40276 C0HRM6 22911602 IC50 = 5 nM T40276 CUN67H 23366085 IC50 = 34000 nM T40276 CLG9Z8 23366090 IC50 = 4400 nM T40276 CW6OB1 23627212 IC50 = 800 nM T40276 CKYB29 23644745 IC50 = 150 nM T40276 C2RV3U 24180608 IC50 > 30000 nM T40276 CK73JS 24742033 Ki = 440 nM T40276 CZKX63 24746470 IC50 = 2200 nM T40276 CKW2O0 24746471 IC50 = 1200 nM T40276 C8QD5W 24746626 IC50 = 2400 nM T40276 C2UOE0 24766030 IC50 > 100000 nM T40276 CJUK39 24770517 IC50 > 50000 nM T40276 CCP2M3 24822704 IC50 > 50000 nM T40276 CM28WD 24825721 IC50 = 22000 nM T40276 CSW5V3 24865437 IC50 = 2000 nM T40276 C5ZM4T 24936119 IC50 > 10000 nM T40276 C4EG8R 24993189 IC50 > 10000 nM T40276 CS3Q8B 24995659 Ki = 260 nM T40276 C1ONA4 24996161 IC50 = 942 nM T40276 C6P1CX 25066843 IC50 = 1600 nM T40276 CDO3X2 25113021 IC50 > 1000 nM T40276 CBI73N 25113026 IC50 > 1000 nM T40276 C1R0JL 25113028 IC50 = 779 nM T40276 C4KL8Q 25113038 IC50 = 961 nM T40276 CV58WZ 25113039 IC50 > 1000 nM T40276 C8KI1Z 25113050 IC50 > 1000 nM T40276 CNG96H 25210579 IC50 > 10000 nM T40276 CD5Z8U 44139091 Ki = 57 nM T40276 CAI56R 44139212 Ki = 76 nM T40276 CNX5R1 44139336 Ki = 15.2 nM T40276 CRD90G 44139337 Ki = 4.1 nM T40276 C4UMB7 44158300 Ki = 89 nM T40276 C4G5DI 44158301 Ki = 3500 nM T40276 CLW80F 44160269 IC50 > 100000 nM T40276 CK73NR 44219749 IC50 > 50000 nM T40276 CIX8V2 44251637 IC50 > 100 nM T40276 C5QFX6 44263382 IC50 = 58 nM T40276 C8RQU2 44263383 IC50 = 36 nM T40276 CZG81D 44263384 IC50 = 1.8 nM T40276 C6YRP1 44263385 IC50 = 1268 nM T40276 C54HZC 44282232 IC50 > 100000 nM T40276 CQ13XB 44291629 Ki = 280 nM T40276 CERT91 44291669 Ki = 36.4 nM T40276 C1FZ6B 44294270 IC50 = 90 nM T40276 C6A9FK 44294365 IC50 = 33 nM T40276 C4HS3C 44294447 IC50 = 3 nM T40276 CFZ31C 44294493 IC50 = 20 nM T40276 C54GFD 44294623 IC50 = 10 nM T40276 CG89DS 44294661 IC50 = 110 nM T40276 CSHC96 44297347 IC50 = 9100 nM T40276 CYF8O6 44297594 IC50 = 2500 nM T40276 CG1Z2B 44303442 IC50 = 70 nM T40276 CNJ63O 44303517 IC50 = 330 nM T40276 C8RJN7 44303745 IC50 = 630 nM T40276 CTM59P 44308069 IC50 = 2 nM T40276 CJ4WB9 44308383 IC50 = 20 nM T40276 C1N6SL 44308409 IC50 = 2500 nM T40276 CO83HF 44308467 IC50 = 2400 nM T40276 CYTA85 44308468 IC50 = 3600 nM T40276 C3M4UP 44308469 IC50 = 220 nM T40276 CY4K5F 44308490 IC50 = 32 nM T40276 C7AG9Y 44308609 IC50 = 3 nM T40276 CYN34A 44308610 IC50 = 5 nM T40276 C79WUE 44308611 IC50 = 4 nM T40276 CS63CK 44308612 IC50 = 60 nM T40276 C47BNR 44310732 IC50 = 10 nM T40276 C2ACB1 44310758 IC50 = 40 nM T40276 CXVB19 44310795 IC50 = 30 nM T40276 CD8OF2 44311036 IC50 = 17 nM T40276 C13TNU 44315122 IC50 = 360 nM T40276 C3YN1R 44315123 IC50 = 710 nM T40276 CPJ57U 44315124 IC50 = 60 nM T40276 C9HA8T 44315171 IC50 = 20 nM T40276 C2T3VN 44315184 IC50 = 80 nM T40276 C3SP0H 44315423 IC50 = 680 nM T40276 C8OAE9 44315457 IC50 = 330 nM T40276 C3JS6X 44315503 IC50 = 30 nM T40276 CEZ68T 44315545 IC50 = 2700 nM T40276 C73MZU 44322457 IC50 = 26000 nM T40276 C2C3MV 44322458 IC50 = 7600 nM T40276 CA4R8N 44322474 IC50 = 25000 nM T40276 C2WUL9 44322520 IC50 = 38000 nM T40276 CU10GA 44322569 IC50 = 110 nM T40276 C3DY4L 44322570 IC50 = 50 nM T40276 C3UMR9 44322571 IC50 = 330 nM T40276 CE0QG3 44322667 IC50 = 3500 nM T40276 C31QSE 44322668 IC50 = 1300 nM T40276 CIB64S 44322669 IC50 = 8000 nM T40276 C42OZF 44322670 IC50 = 800 nM T40276 CPL9E5 44322671 IC50 > 5000 nM T40276 C17GFI 44322684 IC50 = 117000 nM T40276 CG2SL8 44322685 IC50 = 290 nM T40276 CU8CK7 44322686 IC50 = 124000 nM T40276 COCR18 44322713 IC50 = 3700 nM T40276 C6DHT8 44322714 IC50 > 150000 nM T40276 CK7CJ9 44322718 IC50 = 4500 nM T40276 C3VA0L 44322719 IC50 = 2700 nM T40276 C6Z9XL 44322720 IC50 > 50000 nM T40276 C8NR7B 44322740 IC50 = 13000 nM T40276 C4X3UE 44322741 IC50 > 150000 nM T40276 C1JY5B 44322762 IC50 > 150000 nM T40276 CGK4V2 44322763 IC50 = 30 nM T40276 CP2X6J 44322771 IC50 = 24000 nM T40276 CA27PF 44322772 IC50 = 2100 nM T40276 C4P5HM 44322773 IC50 = 9500 nM T40276 CZ7N8D 44322811 IC50 = 5600 nM T40276 C4J3RI 44322813 IC50 = 260 nM T40276 C7WZ4D 44322814 IC50 = 4800 nM T40276 CYDA76 44322815 IC50 > 50000 nM T40276 CI6R4S 44322889 IC50 > 150000 nM T40276 CP6Q9H 44322954 IC50 > 50000 nM T40276 C48NJC 44322981 IC50 = 260 nM T40276 C6K5TE 44322982 IC50 > 150000 nM T40276 CFMB02 44323003 IC50 = 40000 nM T40276 CLPC42 44334296 IC50 = 140 nM T40276 CF61IT 44334334 IC50 = 10 nM T40276 C50EFS 44334355 IC50 = 250 nM T40276 CH9SF8 44334367 IC50 = 110 nM T40276 C3BFI4 44334443 IC50 = 19 nM T40276 CKD2B8 44337790 IC50 > 150000 nM T40276 COJ73E 44355185 Ki = 1.42 nM T40276 CIH03D 44366053 IC50 = 340 nM T40276 CO28BT 44376126 Ki = 2.23 nM T40276 C8X0WA 44384580 Ki = 593 nM T40276 CC95JU 44385548 IC50 = 500 nM T40276 CGQ57L 44386180 IC50 < 25 nM T40276 CI0Y5L 44386181 IC50 = 40 nM T40276 C1W6NC 44386587 IC50 = 10 nM T40276 C0PU3I 44386588 IC50 = 170 nM T40276 C3J6ZO 44386589 IC50 = 60 nM T40276 C4MZI9 44386931 IC50 = 37000 nM T40276 C8B1LV 44394308 IC50 = 17 nM T40276 C4UR6L 44394355 IC50 = 2 nM T40276 C9CX5A 44394369 IC50 = 23 nM T40276 C2PEU9 44394376 IC50 = 480 nM T40276 C8E6JK 44394377 IC50 = 249 nM T40276 C2K9IX 44394397 IC50 = 2187.76 nM T40276 CC34NS 44394398 IC50 = 151 nM T40276 CWUZ78 44394427 IC50 = 198 nM T40276 C4DMA9 44394428 IC50 = 758.58 nM T40276 C8W0DH 44394439 IC50 > 10000 nM T40276 CKCW90 44394463 IC50 = 28 nM T40276 CA7ZI5 44394482 IC50 = 15 nM T40276 CXG8T5 44394503 IC50 = 1450 nM T40276 C5I9QF 44394510 IC50 = 2863 nM T40276 CP9CT3 44394511 IC50 = 41 nM T40276 CFX48I 44394512 IC50 = 30.2 nM T40276 CS83VP 44394536 IC50 = 12.02 nM T40276 CIY32A 44394554 IC50 = 15 nM T40276 C6EZ8Y 44394557 IC50 = 10 nM T40276 CSBC59 44396134 IC50 = 370 nM T40276 CW3BP8 44398371 IC50 > 100000 nM T40276 CY87UN 44456923 Ki = 127 nM T40276 CW0T1S 44456924 Ki = 1100 nM T40276 CS2CV1 44456938 Ki = 88 nM T40276 C5WL1F 44473009 IC50 = 2500 nM T40276 CEG1S5 44473011 IC50 = 2300 nM T40276 C46OMR 44473016 IC50 = 1400 nM T40276 C3VRO9 44557921 IC50 > 10000 nM T40276 C3HW7L 44570553 IC50 > 30000 nM T40276 C17PVE 44570554 IC50 = 2000 nM T40276 CLOY92 44570599 IC50 > 30000 nM T40276 CK06LT 44570600 IC50 > 30000 nM T40276 CJY8S0 44570884 IC50 = 22000 nM T40276 C1S8MC 44575685 IC50 > 150000 nM T40276 CV5GD1 44589002 IC50 = 680 nM T40276 C83KEG 44589022 IC50 = 2660 nM T40276 CU3RF1 45139989 IC50 > 10000 nM T40276 CQGZ06 45139991 IC50 > 10000 nM T40276 CC95PQ 45375865 IC50 = 41000 nM T40276 CEOQ27 45375866 IC50 > 50000 nM T40276 C5S8MA 45485083 IC50 = 1300 nM T40276 CW42YX 45487634 IC50 = 2500 nM T40276 C96BNW 46179972 IC50 > 60000 nM T40276 CYT37A 46232443 IC50 > 50000 nM T40276 C48ZVW 46232555 IC50 > 50000 nM T40276 CS9B1U 46232556 IC50 > 50000 nM T40276 C7ON5A 46233287 IC50 > 10000 nM T40276 CQW97N 46846072 IC50 = 700 nM T40276 CO3P0J 46866604 IC50 < 50000 nM T40276 CSA46L 46874537 IC50 = 6900 nM T40276 CJOM49 46880136 IC50 = 119 nM T40276 CSV5B9 46901859 IC50 = 859 nM T40276 C7YJ2X 46901862 IC50 = 823 nM T40276 C1NKE3 46905987 IC50 = 1400 nM T40276 CE4SU5 47298428 IC50 > 10000 nM T40276 CHSF07 49806372 IC50 > 1000 nM T40276 C5ME3S 49806721 IC50 > 50000 nM T40276 C9L3XR 49838879 IC50 > 40000 nM T40276 CF91RS 49843531 IC50 > 10000 nM T40276 C2Y6QS 50938552 IC50 > 10000 nM T40276 C9NYP4 51036677 IC50 > 10000 nM T40276 C4WRY3 51037112 IC50 > 10000 nM T40276 CRI28Z 51037948 IC50 > 10000 nM T40276 C8CGM9 51346966 IC50 = 3980 nM T40276 CEQN27 52936621 Ki > 1000 nM T40276 CHP06V 52948258 Ki = 140 nM T40276 CD4H3S 53354074 Ki = 15 nM T40276 CM7P3W 53357328 IC50 > 50000 nM T40276 C8NA4L 53384644 IC50 = 32000 nM T40276 CUY9G2 53473663 IC50 = 5.2 nM T40276 CGQ7F8 53473746 IC50 = 3.8 nM T40276 CI1ZG3 53473747 IC50 = 1.2 nM T40276 C67JHW 53473748 IC50 = 23 nM T40276 C7EW6O 53473749 IC50 = 140 nM T40276 CPH34R 53473750 IC50 > 316 nM T40276 CWH1D4 53473825 IC50 > 316 nM T40276 CM8K2V 53473826 IC50 = 5 nM T40276 C9A8HG 53473827 IC50 = 304 nM T40276 C3A8OT 53473828 IC50 > 316 nM T40276 CLX31Q 53473829 IC50 = 48 nM T40276 C8Y9RE 53473918 IC50 = 6.5 nM T40276 C1XFN0 53473919 IC50 = 7.7 nM T40276 CN34UO 53473920 IC50 = 6 nM T40276 C2RE5M 53473921 IC50 = 0.2 nM T40276 C9ZUL0 53473922 IC50 = 5.1 nM T40276 CG6FD5 53474007 IC50 = 7.8 nM T40276 C0Q7JS 53474008 IC50 = 22 nM T40276 C31WZB 53474009 IC50 = 1.4 nM T40276 CJF1M2 53630890 Ki = 0.5 nM T40276 CCM71K 54669828 Ki = 730 nM T40276 CE1ZK6 54759168 IC50 > 10000 nM T40276 CNB76L 56643505 IC50 = 378 nM T40276 C1LZI4 57969746 Ki = 1700 nM T40276 CVK0G4 58056356 IC50 > 50000 nM T40276 COH41P 58325285 IC50 = 410 nM T40276 CJ6ZT2 59332810 IC50 > 1000 nM T40276 C1MR8Q 60097495 IC50 > 10000 nM T40276 CNL04P 60155126 Ki = 15 nM T40276 C56PUM 60155209 Ki = 12 nM T40276 CUJ28O 67112053 IC50 = 20000 nM T40276 C2ZJC1 67113434 IC50 = 16300 nM T40276 CV63UL 67240318 IC50 > 10000 nM T40276 CF39DV 68596931 IC50 = 865 nM T40276 C9XLB3 68597337 IC50 = 661 nM T40276 CMQ58W 68597501 IC50 > 1000 nM T40276 CEZU83 68611347 IC50 > 1000 nM T40276 CJ8G3H 68682755 IC50 = 3.3 nM T40276 CJGH31 70285522 IC50 > 1000 nM T40276 CPZ4F6 71451107 IC50 > 1000 nM T40276 C5RKX0 71452928 IC50 > 1000 nM T40276 CLZ67D 71456431 IC50 > 1000 nM T40276 CS89CL 71456432 IC50 > 1000 nM T40276 CPIH21 71460129 IC50 > 1000 nM T40276 C69NCX 71461845 IC50 > 1000 nM T40276 C9QB5V 71461846 IC50 > 1000 nM T40276 C6O8KG 71461847 IC50 > 1000 nM T40276 CCN01X 71547862 IC50 > 10000 nM T40276 CU60JG 71718528 IC50 > 50000 nM T40276 CV70GZ 71728100 Ki = 1.5 nM T40276 C7Q0AD 76286479 IC50 = 87 nM T40276 CZF0N7 76287389 IC50 = 1500 nM T40276 C28STM 76287526 IC50 = 520 nM T40276 CK25NC 76308133 IC50 = 7.9 nM T40276 C7PKB3 76308134 IC50 = 4.074 nM T40276 CS4JO1 76311726 IC50 = 2.4 nM T40276 C8S4UO 76311727 IC50 = 5 nM T40276 CLZ4V5 76311728 IC50 = 2.239 nM T40276 CGU64E 76315295 IC50 = 2 nM T40276 CG2QS6 76315296 IC50 = 25 nM T40276 CG6AP5 76315297 IC50 = 6.026 nM T40276 C1UN3T 76318975 IC50 = 8.128 nM T40276 CT04LV 76318976 IC50 = 6 nM T40276 C5Q2OW 76322621 IC50 = 4 nM T40276 COQ8H3 76326206 IC50 = 32 nM T40276 CH32FJ 76329809 IC50 = 14 nM T40276 C28MOR 76329810 IC50 = 17.38 nM T40276 CHLN34 76329811 IC50 = 8 nM T40276 CR95LT 76333464 IC50 = 4 nM T40276 CY0UC4 90645194 IC50 > 10000 nM T40276 C0Y8ZK 91933875 IC50 > 10 nM T40276 CY7BI2 118706214 IC50 > 10000 nM T40276 CS12RU 127031435 IC50 = 9200 nM T40276 C2ZD8S 127032024 IC50 > 10000 nM T40276 CO47QJ 133054002 IC50 = 36 nM T40276 CW0P1Q 135433657 IC50 = 3381 nM T40276 CHA4N2 136013680 IC50 > 10 nM T40276 C39NGD 136026545 IC50 > 50000 nM T40276 CZ7EX0 136183413 IC50 > 30000 nM T40276 C1YUD0 136219394 IC50 > 10 nM T40276 CIU8W3 136254389 IC50 > 10 nM T40276 C12UXT 137640959 IC50 = 60 nM T40276 CH15QZ 137643717 IC50 = 2 nM T40276 CUG6N7 137660315 IC50 = 3.1 nM T40276 C6QA5D 137661222 IC50 = 41 nM T40276 C6VB3O 145925651 IC50 >= 5000 nM T40276 C2MD1Q 155513187 IC50 > 10000 nM T40276 D02KPV 37783 Ki = 1.8 nM T40276 D02XHC 448912 IC50 > 100000 nM T40276 D02ZWX 46877400 IC50 = 1500 nM T40276 D03DZO 11715767 IC50 > 10000 nM T40276 D04AXH 11574614 Ki > 10000 nM T40276 D04NGS 5330790 IC50 > 100000 nM T40276 D05KJY 72326 IC50 > 150000 nM T40276 D06ZCX 10455969 IC50 = 32 nM T40276 D07MMG 46877395 IC50 = 1200 nM T40276 D07OAT 456214 IC50 > 10000 nM T40276 D08GIG 46877396 IC50 = 320 nM T40276 D08HFG 24809764 IC50 = 3700 nM T40276 D08JPU 3501 IC50 = 6.2 nM T40276 D09HVH 135566652 IC50 > 10 nM T40276 D0A5YR 46877398 IC50 = 10000 nM T40276 D0D6MH 11617559 IC50 > 13000 nM T40276 D0F0AX 135413546 IC50 = 1200 nM T40276 D0F3XS 46877392 IC50 = 140 nM T40276 D0H7DQ 6419755 IC50 = 21 nM T40276 D0K5ZY 105000 Ki = 6.1 nM T40276 D0KZ2I 46877402 IC50 = 27000 nM T40276 D0L8HO 2399 IC50 = 212 nM T40276 D0QS6O 46877390 IC50 = 270 nM T40276 D0RC8H 46877391 IC50 = 2800 nM T40276 D0T8NU 16757525 IC50 = 1149 nM T40276 D0TO6S 2396 IC50 = 1.6 nM T40276 D0V3TE 46877397 IC50 = 3000 nM T40276 D0X2DH 17814743 IC50 = 223 nM T85467 D05ZTH 5311181 Ki = 3700 nM T85467 D06FEA 5280360 Ki = 0.33 nM T85467 D0WL5V 9867642 Ki = 892 nM T85467 D00HTY 5280363 IC50 = 322 nM T85467 D00IQH 11677589 Ki > 5000 nM T85467 D00MZK 9911469 Ki = 8200 nM T85467 D00SOZ 44230999 IC50 > 10000 nM T85467 D01SHJ 56944705 IC50 > 10000 nM T85467 D08QWQ 5283081 EC50 = 8600 nM T85467 D0G6EI 9890801 Ki > 2800 nM T85467 D0K1EG 11508736 IC50 > 10000 nM T85467 D0M4TJ 44219292 Ki = 143 nM T85467 D0SP5V 49843471 IC50 > 25000 nM T85467 D0Y3LL 18376177 Ki > 3200 nM T85467 D0W2OT 5311035 Ki > 10000 nM T85467 D02RUO 9807448 Ki > 10000 nM T85467 D08QHS 11296282 IC50 = 4.6 nM T85467 C5Z8HC 132836 Ki = 82 nM T85467 CAZT67 1283333 Ki = 794.33 nM T85467 C4P2CZ 1450040 Ki = 1000 nM T85467 C6DSA1 1450080 Ki = 158.49 nM T85467 C2JB5D 1450082 Ki = 630.96 nM T85467 CO1IZ6 1450090 Ki = 3162.28 nM T85467 CI45ZG 1450104 Ki = 1000 nM T85467 CO8A9R 1450111 Ki = 316.23 nM T85467 CANV86 1498200 Ki > 5000 nM T85467 C3LM8E 1498314 Ki > 5000 nM T85467 CLM8P6 2114670 Ki = 79.43 nM T85467 C0L6YE 3231721 Ki = 794.33 nM T85467 C2XLU7 5311228 Ki = 2700 nM T85467 CK16QC 5311234 IC50 = 186 nM T85467 CO7N1Z 5311239 IC50 > 10000 nM T85467 CZ15QS 6441607 EC50 = 2000 nM T85467 CC9BE3 6443852 EC50 = 4.1 nM T85467 CZA41R 9808508 Ki = 2800 nM T85467 C6TA3N 9809136 Ki = 4000 nM T85467 CV24TI 9817292 Ki = 80 nM T85467 CF6Y2K 9820333 IC50 > 3200 nM T85467 CYNX09 9825293 EC50 > 20000 nM T85467 C5J8WP 9830442 Ki = 51200 nM T85467 CG3IS9 9830839 Ki = 7000 nM T85467 C9IV7J 9844175 IC50 < 3162.28 nM T85467 C97MIQ 9865111 Ki = 65 nM T85467 C6V1BA 9872741 Ki = 6000 nM T85467 CA2I4Z 9873528 Ki = 2400 nM T85467 CKMW12 9874010 Ki = 5000 nM T85467 C38DYF 9885106 Ki = 1900 nM T85467 CF0HC5 9888589 IC50 > 10000 nM T85467 CFC8G4 9894720 Ki > 3000 nM T85467 CA5N0K 9895436 Ki = 16000 nM T85467 CQ0X9R 9909510 IC50 > 10000 nM T85467 CBY0I3 9913176 Ki = 2.1 nM T85467 C7MA6V 9916766 Ki = 13000 nM T85467 CN2UX4 9938625 Ki = 3600 nM T85467 CICE70 9938626 Ki = 5000 nM T85467 C1KAC5 9938669 Ki = 4700 nM T85467 C6DQ3W 9938995 Ki = 2200 nM T85467 CWDT69 9939791 Ki = 1300 nM T85467 CWS81C 9944231 Ki = 750 nM T85467 C4Q7RI 9953337 Ki = 5 nM T85467 C6SGH7 9954562 Ki = 1.1 nM T85467 C4UK2Q 9955802 Ki > 3000 nM T85467 C6ZM4U 9959673 Ki = 1200 nM T85467 CCD30P 9960839 Ki > 100000 nM T85467 C4Z7BL 9965922 Ki = 10 nM T85467 C5AF0B 9975502 Ki = 10000 nM T85467 CZUJ52 10001608 IC50 = 3700 nM T85467 CCD24K 10007859 Ki = 501.19 nM T85467 CQ3GW6 10047541 IC50 = 1000 nM T85467 CNE21V 10095268 Ki = 501.19 nM T85467 COR8X7 10109445 Ki > 100000 nM T85467 C6UI2Z 10111602 Ki = 8 nM T85467 CBYV78 10112486 Ki = 520 nM T85467 C93DSI 10113454 Ki = 38000 nM T85467 C1J6DM 10113842 Ki = 153 nM T85467 C26QRM 10118889 Ki = 27 nM T85467 C98DZA 10127780 IC50 < 3162.28 nM T85467 CS9R6Z 10127791 IC50 < 3162.28 nM T85467 C1QI8X 10128061 IC50 < 3162.28 nM T85467 C1YW6D 10139917 Ki = 17 nM T85467 C6BOW4 10144273 Ki = 120 nM T85467 CWN91Y 10150770 IC50 < 3162.28 nM T85467 CCPI72 10151282 IC50 < 3162.28 nM T85467 C28CIN 10152107 IC50 < 3162.28 nM T85467 C6W9IC 10158725 Ki = 23 nM T85467 CM3SE6 10168694 Ki = 16 nM T85467 C6Y3CX 10173065 IC50 < 3162.28 nM T85467 C3FXN2 10174660 IC50 < 3162.28 nM T85467 C71GVU 10178073 Ki = 7 nM T85467 CEM21G 10181606 Ki = 25 nM T85467 CU47VL 10194556 IC50 < 3162.28 nM T85467 C2MEG8 10195119 IC50 < 3162.28 nM T85467 CZKM14 10195696 IC50 < 3162.28 nM T85467 C6X5CP 10202765 Ki = 13000 nM T85467 C4Y9RW 10215735 IC50 < 3162.28 nM T85467 CNRP47 10216080 IC50 < 3162.28 nM T85467 CRA06V 10216528 IC50 < 3162.28 nM T85467 CW13VB 10216958 IC50 < 3162.28 nM T85467 CP8KN7 10227492 Ki = 21 nM T85467 C6FM0Z 10238855 IC50 < 3162.28 nM T85467 C0ED9Y 10251023 IC50 > 10000 nM T85467 C89CXB 10271490 Ki = 13 nM T85467 COFP92 10275762 Ki = 6.7 nM T85467 CV7H2E 10275911 IC50 > 3200 nM T85467 CL7YG3 10287121 Ki > 13000 nM T85467 CP6D2N 10288374 IC50 < 3162.28 nM T85467 C40QFO 10291963 Ki = 11000 nM T85467 CV9QL7 10302378 Ki = 0.6 nM T85467 CL65HU 10310187 IC50 < 3162.28 nM T85467 CRM34S 10311325 IC50 < 3162.28 nM T85467 C3C5IM 10322469 Ki = 38000 nM T85467 C51JIX 10389527 EC50 > 20000 nM T85467 CB19MW 10402929 Ki = 32 nM T85467 CI5HA0 10648334 IC50 > 10000 nM T85467 C9YQG5 10670992 IC50 > 10000 nM T85467 C7GY6X 10739351 IC50 > 10000 nM T85467 CY8IB2 10740699 IC50 > 10000 nM T85467 C12SBH 10741017 IC50 > 10000 nM T85467 CG17HE 10741197 IC50 > 10000 nM T85467 CKST02 11122314 IC50 > 10000 nM T85467 CEI08Z 11155228 Ki = 3 nM T85467 CC8PQ2 11156167 EC50 = 7.4 nM T85467 CF6EO3 11210487 Ki = 1400 nM T85467 C4S5MX 11249458 Ki > 10000 nM T85467 C70ESM 11269563 Ki = 1200 nM T85467 COS4C2 11294085 EC50 = 0.7 nM T85467 C9E4SW 11294166 Ki > 20000 nM T85467 CFDA92 11326896 IC50 > 3200 nM T85467 CIM8K7 11328569 EC50 = 25 nM T85467 CQU62G 11337782 Ki = 77000 nM T85467 C4IK7Y 11339240 Ki > 100000 nM T85467 CQ7Z5B 11339406 IC50 > 3200 nM T85467 CBP71Y 11362836 EC50 = 4.7 nM T85467 CN2TG7 11387144 Ki > 3000 nM T85467 CUWE27 11405770 Ki = 90300 nM T85467 CXPO04 11408533 Ki > 20000 nM T85467 CP4LS0 11440167 Ki = 79000 nM T85467 CZ4K0P 11476788 Ki = 5063 nM T85467 CM6Z1E 11486771 IC50 > 3200 nM T85467 CE2JA4 11488860 Ki = 830 nM T85467 CW3YO5 11494768 IC50 > 25000 nM T85467 CQ6IU7 11509269 IC50 > 10000 nM T85467 CS2LR0 11516353 IC50 > 25000 nM T85467 CF2OM8 11539410 IC50 > 25000 nM T85467 CM7HK0 11551847 IC50 > 25000 nM T85467 CJ2OE0 11575201 IC50 > 20000 nM T85467 C1W2ZK 11577792 Ki > 6000 nM T85467 C7Y6XJ 11597294 Ki = 470 nM T85467 C2M8HZ 11610353 IC50 > 25000 nM T85467 CGS72I 11618662 IC50 > 20000 nM T85467 C9L5VD 11631813 IC50 > 25000 nM T85467 CD7R5P 11631965 IC50 > 25000 nM T85467 CMB6F9 11653874 IC50 > 25000 nM T85467 CB7SR6 11657311 IC50 = 10 nM T85467 C51UDK 11667741 IC50 > 10000 nM T85467 CAL96X 11683088 IC50 > 20000 nM T85467 CW8RY9 11689895 IC50 > 25000 nM T85467 C9CM2R 11695689 IC50 > 10000 nM T85467 C3BSV4 11696697 Ki = 3340 nM T85467 CNYK74 11743212 Ki = 3 nM T85467 CK2EZ6 11962967 Ki < 10000 nM T85467 CH26TZ 11963255 Ki < 10000 nM T85467 CR82PA 12112238 Ki = 84 nM T85467 CX0M2W 12112239 Ki = 340 nM T85467 C32GBT 12137443 Ki = 54000 nM T85467 C93FZV 13174090 EC50 = 0.89 nM T85467 CT34LO 13230981 Ki = 419 nM T85467 CO19GA 14372497 Ki > 300 nM T85467 CB1N7G 14429703 EC50 = 0.34 nM T85467 C06OGJ 15486805 IC50 = 5900 nM T85467 C0L3VU 15486806 IC50 > 10000 nM T85467 CU5J6N 15491229 Ki > 100000 nM T85467 CMG0Z1 15491230 Ki > 100000 nM T85467 CWQ8B9 15551228 Ki = 0.7 nM T85467 CZ87CN 15907747 Ki = 1600 nM T85467 CVEO28 15907748 Ki = 4700 nM T85467 CIS83K 15947857 Ki = 2700 nM T85467 C3L0RK 15948325 Ki = 4000 nM T85467 CRT3I2 15979081 EC50 = 2.7 nM T85467 CI61TE 16678098 IC50 > 10000 nM T85467 CK68XW 18196125 Ki > 25118.86 nM T85467 CS8M2G 18973764 Ki = 2300 nM T85467 CX08BC 21198692 Ki = 3.2 nM T85467 CR37AJ 21362845 Ki = 110 nM T85467 C6UT1I 21362849 Ki = 820 nM T85467 C4IFY8 21362851 Ki = 55 nM T85467 C9HQN0 21362853 Ki = 89 nM T85467 C6F8QI 21362863 Ki = 1500 nM T85467 CL5O9E 21362867 Ki = 240 nM T85467 C58NCB 21362869 Ki = 5900 nM T85467 CHS9L6 21362879 Ki = 27 nM T85467 CW7R1M 21362893 Ki = 53 nM T85467 C9HD2W 21362900 Ki = 46 nM T85467 CSUO46 21362905 Ki = 620 nM T85467 CJ65SZ 21362910 Ki = 590 nM T85467 CFV24G 21362912 Ki = 200 nM T85467 C0UT6R 22008966 Ki = 2.4 nM T85467 CJ4M7P 22008967 Ki = 2.4 nM T85467 C9TSB7 22009003 Ki = 9 nM T85467 C8SON3 22009004 Ki = 1.6 nM T85467 CAML12 22009006 Ki = 5 nM T85467 C5DGQ4 22009008 Ki = 1.6 nM T85467 C5SJ2H 22009011 Ki = 10 nM T85467 C3D2LR 22990263 Ki = 1600 nM T85467 CF81SW 23582412 IC50 > 10000 nM T85467 CP2S4J 23663736 Ki = 3200 nM T85467 C9H4WT 23686961 Ki = 1995.26 nM T85467 CASU54 23696973 IC50 = 1258.93 nM T85467 C42LYP 24765153 Ki = 710 nM T85467 CF72YI 24765671 Ki >= 785 nM T85467 C31JZP 24765672 Ki >= 2500 nM T85467 C4QX7Y 24765675 Ki >= 930 nM T85467 CL7Z9U 24765768 Ki >= 110 nM T85467 C0R6TW 24784836 Ki = 1000 nM T85467 CFQA40 24952577 Ki > 7282 nM T85467 CD98IN 24952580 Ki > 456 nM T85467 C81WVN 24952927 Ki > 5474 nM T85467 CZT83E 24952928 Ki > 501 nM T85467 C8YHX3 24953283 Ki > 224 nM T85467 CZ93FO 24953285 Ki > 628 nM T85467 C17JTY 24953286 Ki > 2226 nM T85467 CFT0W5 24953624 Ki > 4992 nM T85467 C42VMD 24953625 Ki > 3461 nM T85467 C7B2EW 24953628 Ki > 2117 nM T85467 CXQJ67 25002382 Ki >= 1291 nM T85467 CN5SH9 25003075 Ki = 7400 nM T85467 C8CH5S 25181432 IC50 = 0.3 nM T85467 C13DMB 25181438 IC50 = 1 nM T85467 C4J2BS 25195248 IC50 = 3.5 nM T85467 CR10FW 30897313 IC50 = 23000 nM T85467 C3LQ4B 44129707 IC50 = 9.2 nM T85467 CNOF71 44138108 Ki = 851 nM T85467 CSRV98 44157014 IC50 = 7.4 nM T85467 C2AV1K 44190762 IC50 = 1220 nM T85467 C2O0NL 44230575 IC50 > 10000 nM T85467 CQ13MH 44234032 Ki = 210 nM T85467 CR68BA 44250281 Ki = 1.259 nM T85467 C3RM7D 44250282 Ki = 7.943 nM T85467 CN90FE 44269464 Ki = 2315 nM T85467 C1L0ET 44269468 Ki > 13000 nM T85467 C5KRQ4 44269486 Ki = 700 nM T85467 CL6M2P 44269516 Ki = 2000 nM T85467 CON8R9 44269520 Ki > 13000 nM T85467 C6MBG0 44269521 Ki > 13000 nM T85467 CZ3Q1L 44269523 Ki > 13000 nM T85467 CRL61O 44269532 Ki > 13000 nM T85467 C1Z4LU 44269540 Ki > 13000 nM T85467 CM72FA 44269542 Ki = 1220 nM T85467 CN0JV2 44269543 Ki > 13000 nM T85467 C28UJH 44269544 Ki > 13000 nM T85467 CR1IY6 44269568 Ki = 10560 nM T85467 CI3C9O 44269596 Ki = 2014 nM T85467 CC0EW9 44269597 Ki > 13000 nM T85467 CWJC89 44285146 IC50 > 10000 nM T85467 C5P9CF 44285208 IC50 > 10000 nM T85467 CCD2S1 44285209 IC50 > 10000 nM T85467 C9U7YH 44285251 IC50 > 10000 nM T85467 C6EZ1R 44285252 IC50 > 10000 nM T85467 CS64GQ 44285310 EC50 > 20000 nM T85467 CDP9F2 44285328 IC50 > 10000 nM T85467 CY37TX 44289792 Ki = 12000 nM T85467 C6JAE2 44289921 Ki = 16000 nM T85467 CDJV85 44289968 Ki = 12000 nM T85467 C68XKV 44289977 Ki = 131000 nM T85467 CHZ21Q 44290257 Ki > 100000 nM T85467 CO31WZ 44290262 Ki > 100000 nM T85467 COF9C2 44290263 Ki > 100000 nM T85467 C4SEW6 44290266 Ki = 8 nM T85467 CEVM85 44290267 Ki = 56000 nM T85467 C7RDN9 44290271 Ki > 100000 nM T85467 CN5RG9 44290272 Ki > 100000 nM T85467 CZ59QY 44290312 Ki > 100000 nM T85467 CAV76T 44290314 Ki = 4900 nM T85467 C4F8YR 44290494 Ki > 100000 nM T85467 CS7RH0 44320126 Ki = 120 nM T85467 CLR9F5 44320272 Ki = 330 nM T85467 CKYS39 44320294 Ki = 610 nM T85467 CH6TK1 44320321 Ki = 440 nM T85467 CYI1O0 44320373 Ki = 740 nM T85467 C0V3OA 44320388 Ki = 150 nM T85467 C01HGT 44320405 Ki = 480 nM T85467 CS58ZQ 44320433 Ki = 510 nM T85467 CS52ZR 44324368 Ki = 4600 nM T85467 CM72WE 44349503 Ki = 16 nM T85467 C9PO1Q 44349528 Ki = 35 nM T85467 C1R7HU 44349531 Ki = 1700 nM T85467 CHO7X0 44349551 Ki = 52 nM T85467 CLN63A 44377464 Ki = 110 nM T85467 CJIS72 44390782 Ki = 19 nM T85467 C43VIA 44390806 Ki = 41 nM T85467 CB8H4V 44390831 Ki = 7 nM T85467 CWL1X4 44400355 Ki > 1000 nM T85467 C76QVA 44402710 Ki > 1900 nM T85467 CRAX23 44402824 Ki > 10000 nM T85467 CYG6Q2 44409742 IC50 > 2000 nM T85467 CKM6S2 44409910 IC50 = 20000 nM T85467 CS42GV 44409918 IC50 > 3200 nM T85467 CIB2W5 44419347 Ki = 3 nM T85467 CF35LY 44419350 Ki = 65 nM T85467 CNK1X9 44419351 Ki = 56 nM T85467 C91JXT 44419374 Ki = 9 nM T85467 CNF4W2 44419379 Ki = 9 nM T85467 CS3IW4 44419380 Ki = 10 nM T85467 CBQ01L 44419384 Ki = 10 nM T85467 C01PQW 44430772 IC50 < 3162.28 nM T85467 CWG71J 44430773 IC50 < 3162.28 nM T85467 C3RGU1 44430774 IC50 < 3162.28 nM T85467 CGS0P7 44442327 Ki = 9000 nM T85467 CF32IP 44442331 Ki = 10000 nM T85467 C8KQP9 44448929 Ki = 398.11 nM T85467 C3UV1I 44448955 Ki = 794.33 nM T85467 C7N1IY 44448984 Ki = 501.19 nM T85467 C94ZPE 44448986 Ki = 316.23 nM T85467 CSA84U 44449089 Ki = 501.19 nM T85467 C3E7YJ 44449112 Ki = 398.11 nM T85467 CDBE16 44450497 Ki > 21360 nM T85467 CUHD74 44564571 IC50 = 12.4 nM T85467 CWB91Y 44564572 IC50 = 15.7 nM T85467 C35GNP 44564573 IC50 = 4.6 nM T85467 CX5F3C 44564647 IC50 = 9.4 nM T85467 CZA96G 44564648 IC50 = 18.4 nM T85467 CL3MA0 44564649 IC50 = 11.8 nM T85467 CZ75IN 44564650 IC50 = 54.1 nM T85467 CO86IB 44564685 IC50 = 8.7 nM T85467 C0D2LM 44564686 IC50 = 3.5 nM T85467 CH7RI1 44564687 IC50 = 6.5 nM T85467 C9YA2K 44564723 IC50 = 5.9 nM T85467 CB5HU0 44564724 IC50 = 44.9 nM T85467 CRP29C 44564725 IC50 = 17.5 nM T85467 C7JK5M 44564726 IC50 = 11.9 nM T85467 C2JZ3V 44564770 IC50 = 1100 nM T85467 CTB9R8 44564771 IC50 = 100.8 nM T85467 CT5DQ8 44564772 IC50 = 5.1 nM T85467 CA05LN 44564804 EC50 = 26.1 nM T85467 CZHR20 44564805 IC50 = 27.3 nM T85467 CR0M4T 44564806 IC50 = 195.9 nM T85467 COF62Z 44564807 IC50 = 18.5 nM T85467 CUZH96 44564840 IC50 = 612.4 nM T85467 C6XE0K 44564841 IC50 = 7.2 nM T85467 CS1ZJ0 44564842 IC50 = 145.8 nM T85467 C9F3WO 44564843 IC50 = 4.4 nM T85467 CU3I1M 44564890 IC50 = 1.9 nM T85467 CE2VG3 44564891 IC50 = 6.1 nM T85467 CND54C 44564892 IC50 = 2.6 nM T85467 C2VR6S 44564893 IC50 = 3.2 nM T85467 CUD1W2 44564934 IC50 = 392.9 nM T85467 CU7C4V 44564935 IC50 = 3.8 nM T85467 C6VK1D 44564936 IC50 = 84.8 nM T85467 C18GXI 44564937 IC50 = 9.7 nM T85467 CZ74GB 44564990 IC50 = 6.7 nM T85467 C0YLB2 44564991 IC50 = 4.4 nM T85467 CTEY20 44564992 IC50 = 316.3 nM T85467 C8WMH6 44564993 IC50 = 5.1 nM T85467 CSHZ25 44565043 IC50 = 8.5 nM T85467 CPCT59 44565044 IC50 = 7.2 nM T85467 C0NF1S 44565193 IC50 = 26.9 nM T85467 C07ODW 44570000 IC50 = 3 nM T85467 CIRO75 44570001 IC50 = 545 nM T85467 CPJR60 44570002 IC50 = 6.1 nM T85467 CI65RQ 44570003 IC50 = 7.6 nM T85467 CCR37Z 44570004 IC50 = 10.7 nM T85467 C3V0XA 44570005 IC50 = 43 nM T85467 C8PW9K 44570036 IC50 = 0.7 nM T85467 C9OKN4 44570047 IC50 = 11.9 nM T85467 C4K0PI 44570147 IC50 = 134 nM T85467 CG48CP 44570148 IC50 = 48.7 nM T85467 CY0DJ5 44570149 IC50 = 3 nM T85467 CO6S3I 44570150 IC50 = 2.3 nM T85467 C6J9CB 44570151 IC50 = 95 nM T85467 CEHZ26 44570152 IC50 = 11.6 nM T85467 CNV72G 44570153 IC50 = 236.2 nM T85467 CC9IU2 44570187 IC50 = 5.7 nM T85467 CLX9P1 44570188 IC50 = 122.1 nM T85467 C07DHR 44570189 IC50 = 2.2 nM T85467 CG6MN5 44570190 IC50 = 0.3 nM T85467 C5YN4M 44570191 IC50 = 11.4 nM T85467 CK51IN 44570192 IC50 = 5 nM T85467 C2BDI7 44570193 IC50 = 14.3 nM T85467 C14BNG 44570194 IC50 = 30 nM T85467 CWZT54 44570230 IC50 = 651 nM T85467 CB0AQ6 44570231 IC50 = 3.6 nM T85467 CXO34D 44570232 IC50 = 2.2 nM T85467 C2H0CS 44570233 IC50 = 36.7 nM T85467 C29VWK 44570234 IC50 = 88.4 nM T85467 COW68J 44570235 IC50 = 16.7 nM T85467 C0DFG4 44570279 IC50 = 0.2 nM T85467 C97CMX 44570280 IC50 = 1.9 nM T85467 C3FB4E 44570281 IC50 = 1.3 nM T85467 C65VON 44570282 IC50 = 24.1 nM T85467 C60YFH 44570313 IC50 = 9.8 nM T85467 CYP9K4 44570314 IC50 = 1.8 nM T85467 CI52EW 44570315 IC50 = 5.8 nM T85467 C1KX3O 44570316 IC50 = 24 nM T85467 C4EOR8 44570353 IC50 = 2.8 nM T85467 C2IVO6 44570354 IC50 = 3.9 nM T85467 CSJ4L9 44570355 IC50 = 37.9 nM T85467 CZE85H 44570398 IC50 = 9.3 nM T85467 CR2U4Q 44570399 IC50 = 3.6 nM T85467 C1GH9U 44570400 IC50 = 3.4 nM T85467 CW9SZ0 44570401 IC50 = 0.5 nM T85467 C4NY9J 44570443 IC50 = 8.2 nM T85467 CQ7GM4 44570444 IC50 = 34 nM T85467 CG5D8Z 44570445 IC50 = 10.5 nM T85467 CFVQ49 44570446 IC50 = 66.1 nM T85467 C2C0TY 44570484 IC50 = 9.4 nM T85467 C9XUQ6 44570485 IC50 = 3.6 nM T85467 C4RUX9 44570486 IC50 = 18.8 nM T85467 C7DH1F 44570523 IC50 = 79.6 nM T85467 CXJN41 44570524 IC50 = 40.2 nM T85467 C0TV4L 44570525 IC50 = 8.8 nM T85467 CQ1TM2 44570562 IC50 = 3.9 nM T85467 C29NBD 44570563 IC50 = 41 nM T85467 C6TO1X 44570564 IC50 = 5.9 nM T85467 CGH38O 44570604 IC50 = 1.7 nM T85467 C6SO3A 44570605 IC50 = 544.4 nM T85467 CPC85Y 44570606 IC50 = 9.2 nM T85467 CLA3X6 44570607 IC50 = 52 nM T85467 C1T3RM 44570638 IC50 = 198 nM T85467 CI63BN 44570639 IC50 = 44.8 nM T85467 CO2SW5 44570640 IC50 = 13.8 nM T85467 CP72CG 44570641 IC50 = 5.7 nM T85467 CP71ZX 44570665 IC50 = 3.4 nM T85467 CJKA53 44570666 IC50 = 9.4 nM T85467 CPH51Y 44570667 IC50 = 2.5 nM T85467 CSW92V 44570668 IC50 = 4.3 nM T85467 CTW6L7 44570712 IC50 = 3.7 nM T85467 C6DK1U 44570827 IC50 = 5.6 nM T85467 C6JO4B 44570828 IC50 = 9.8 nM T85467 CUFQ35 44570829 IC50 = 3.2 nM T85467 CT6IM9 44570870 IC50 = 1.8 nM T85467 CS75YT 44570871 IC50 = 556.9 nM T85467 CQF92X 44570872 IC50 = 29.9 nM T85467 CQ5V1Z 44570910 IC50 = 20.6 nM T85467 C6RQF4 44570911 IC50 = 11.2 nM T85467 CM6V5A 44570912 IC50 = 267.4 nM T85467 CP3TK2 44570950 IC50 = 10.7 nM T85467 C3HW8Q 44570953 IC50 = 314 nM T85467 CK28RM 44570993 IC50 = 261 nM T85467 C1BI2V 44570995 IC50 = 180 nM T85467 CGX17U 44571206 IC50 = 6.8 nM T85467 CWO4P3 44571243 IC50 = 1.7 nM T85467 CLI87C 44571244 IC50 = 2.3 nM T85467 C1OSI9 44571245 IC50 = 2.2 nM T85467 CN42VJ 44571246 IC50 = 9.5 nM T85467 CVF2G5 44571289 IC50 = 3.5 nM T85467 C5URT2 44571290 IC50 = 3.8 nM T85467 CE4UO5 44571291 IC50 = 6.4 nM T85467 C0I6NX 44571292 IC50 = 13.4 nM T85467 C63TLM 44571318 IC50 = 57.2 nM T85467 C7UIO1 44571319 IC50 = 15.2 nM T85467 CSAQ62 44571320 IC50 = 9.2 nM T85467 C1P9ZE 44571321 IC50 = 3.8 nM T85467 CK1GW9 44571352 IC50 = 84.1 nM T85467 CANI83 44571353 IC50 = 5.6 nM T85467 CXQI89 44571354 IC50 = 12.9 nM T85467 C2PIB9 44571355 IC50 = 3.5 nM T85467 CK8Y5R 44594042 IC50 = 3.7 nM T85467 CYCW19 44626787 IC50 = 45 nM T85467 CV06JZ 44626788 IC50 = 98 nM T85467 C5PT0Z 44626877 IC50 = 2 nM T85467 CYS07E 44626878 IC50 = 420 nM T85467 CNP4C2 44626879 IC50 = 5 nM T85467 CD09TJ 44626880 IC50 = 71 nM T85467 C6YJT1 44626881 IC50 = 88 nM T85467 CIR3B4 44626882 IC50 = 14 nM T85467 CP3NT6 44626975 IC50 = 14.2 nM T85467 C4SH2N 44626976 IC50 = 25 nM T85467 CBSH12 44626977 IC50 = 2710 nM T85467 C0NIO8 44626978 IC50 = 326 nM T85467 COD4F6 44626979 IC50 = 34 nM T85467 C56OQV 44626980 IC50 = 4044 nM T85467 CF7X3J 44627070 IC50 = 10091 nM T85467 CMF94N 44627071 IC50 = 2.5 nM T85467 CHGN39 44627072 IC50 = 2.7 nM T85467 C1WV7T 44627073 IC50 = 2.4 nM T85467 C0I2UV 44627074 IC50 = 2.5 nM T85467 CRD80U 44627172 IC50 = 2838 nM T85467 CH0NT4 44627173 IC50 = 1146 nM T85467 CRV89Z 44627174 IC50 = 2.2 nM T85467 C2R3UC 44627175 IC50 = 3 nM T85467 CE2PR6 44627282 IC50 = 8.9 nM T85467 CF28KZ 44627283 IC50 = 1552 nM T85467 CUA1I8 44627284 IC50 = 27 nM T85467 C9Y6HL 44627285 IC50 = 27.6 nM T85467 C8DXC6 44627286 IC50 = 89.5 nM T85467 CQIK27 44627395 IC50 = 1.1 nM T85467 CB2WF8 44627396 IC50 = 65.7 nM T85467 CQ8SU1 44627397 IC50 = 4.9 nM T85467 CQE52R 44627398 IC50 = 14.6 nM T85467 CBTA12 44627399 IC50 = 14 nM T85467 C9R5PA 44627513 IC50 = 6.6 nM T85467 C4W1ZG 44627515 IC50 = 7 nM T85467 CJG7N1 44627621 IC50 = 2 nM T85467 CT2JH9 44627622 IC50 = 13.8 nM T85467 CQA6S3 44627718 IC50 = 1 nM T85467 C83LNC 44627719 IC50 = 14.5 nM T85467 C7ZJO3 44627720 IC50 = 393 nM T85467 CQ0YU8 44627721 IC50 = 46.4 nM T85467 CD7XR3 44627829 IC50 = 501 nM T85467 CLI8D4 44627830 IC50 = 2045 nM T85467 CM7X6Z 45267483 Ki = 199.53 nM T85467 CI93EW 45267497 Ki = 199.53 nM T85467 C8F4YQ 45267514 Ki = 794.33 nM T85467 CW94TZ 45268367 Ki = 100 nM T85467 CD39KU 45268368 Ki = 199.53 nM T85467 C41RIZ 45268369 Ki = 15.85 nM T85467 C69GNM 45269218 Ki = 158.49 nM T85467 CB62SZ 45269223 Ki = 19.95 nM T85467 CJQ94Y 45269232 Ki = 25.12 nM T85467 CDM6S1 45269240 Ki = 1995.26 nM T85467 CL48SF 45270083 Ki = 3.162 nM T85467 C3SK7A 45270084 Ki = 630.96 nM T85467 C94IWH 45270915 Ki = 12.59 nM T85467 CW36LH 45270922 Ki = 12.59 nM T85467 CMAY-54 45271758 Ki > 25118.86 nM T85467 C0SX7L 45271759 Ki = 398.11 nM T85467 C8KFW0 45271767 Ki = 5.012 nM T85467 CI4B1Z 45272630 Ki = 1258.93 nM T85467 CO4X6P 45272639 Ki = 1.259 nM T85467 C2O9HS 45273534 Ki = 501.19 nM T85467 C2T9FV 45488088 IC50 = 7200 nM T85467 C6QD3H 45488089 IC50 = 6400 nM T85467 C3BI4N 45488090 IC50 = 34860 nM T85467 CLV46P 45488091 IC50 = 5950 nM T85467 C1U0NY 45488094 IC50 = 6490 nM T85467 CP5B3C 45488095 IC50 = 17710 nM T85467 C6KC8G 45488096 IC50 = 3 nM T85467 CKY7W8 45488100 IC50 = 1.3 nM T85467 C5AY6M 46220498 Ki > 5000 nM T85467 CH0Z3G 46879718 IC50 = 2 nM T85467 C02OTI 46879719 IC50 = 24 nM T85467 C0VMT5 46879756 IC50 = 59 nM T85467 CVF7D1 46879757 IC50 = 5 nM T85467 CM89HE 46879758 IC50 = 1 nM T85467 CV7T3D 46879759 IC50 = 1978 nM T85467 CND97E 46879800 IC50 = 8 nM T85467 C3R0ZV 46879801 IC50 = 3 nM T85467 CN3DA1 46879802 IC50 = 2 nM T85467 CB9RN4 46879858 IC50 = 11 nM T85467 C7XP6O 46879859 IC50 = 1 nM T85467 CFQT59 46879860 IC50 = 4 nM T85467 CS4F0X 46879894 IC50 = 1 nM T85467 CPH53K 46879895 IC50 = 1 nM T85467 C61SDT 46879896 IC50 = 20 nM T85467 CTG6P5 46879998 IC50 = 12 nM T85467 C9GZP5 46879999 IC50 = 44 nM T85467 CTR35I 46880000 IC50 = 664 nM T85467 CK68VO 46880001 IC50 = 1315 nM T85467 C2B6IK 46880037 IC50 = 1020 nM T85467 CC7ZB2 46880038 IC50 = 363 nM T85467 C6E2UQ 46880039 IC50 = 244 nM T85467 CSE91V 46880040 IC50 = 2570 nM T85467 C79HSW 46880091 IC50 = 17850 nM T85467 C5FET9 46885340 IC50 = 5 nM T85467 CH9M2P 46885341 IC50 = 2.9 nM T85467 CI6K8H 46885342 IC50 = 56 nM T85467 C78XQT 46885343 IC50 = 0.5 nM T85467 C0J4TA 46885384 IC50 = 0.2 nM T85467 C6LY9A 46885385 IC50 = 0.7 nM T85467 C6JB3C 46885386 IC50 = 1.2 nM T85467 CC7XA6 46885387 IC50 = 1.3 nM T85467 C49QGD 46885431 IC50 = 23.6 nM T85467 C8F7JR 46885432 IC50 = 0.3 nM T85467 CNMS56 46885433 IC50 = 0.4 nM T85467 CG9BA8 46885434 IC50 = 0.5 nM T85467 C9KT8F 46885501 IC50 = 0.6 nM T85467 CP2NF6 46885502 IC50 = 0.9 nM T85467 CX7YK8 46885503 IC50 = 55.4 nM T85467 CI3O9E 46885504 IC50 = 35.5 nM T85467 CC20YM 46885538 IC50 = 0.7 nM T85467 C5QN0E 46885539 IC50 = 0.4 nM T85467 C42ZNY 46885540 IC50 = 243.1 nM T85467 CP09TQ 46885541 IC50 = 186.9 nM T85467 CN47XP 46885575 IC50 = 45.4 nM T85467 CX0Y8P 46885576 IC50 = 3.8 nM T85467 CI2Q5J 46885577 IC50 = 13 nM T85467 CE5BF8 46885602 IC50 = 660 nM T85467 C4STZ3 46885603 IC50 = 23.9 nM T85467 CXO8P5 46885604 IC50 = 3.3 nM T85467 CR0DB6 46885605 IC50 = 82.4 nM T85467 C49DSC 46885606 IC50 = 6.5 nM T85467 C7IJ0G 46885649 IC50 = 9.8 nM T85467 C3QT8M 46885650 IC50 = 0.5 nM T85467 C6QSN0 46885651 IC50 = 0.5 nM T85467 CM20ZL 46885652 IC50 = 3.5 nM T85467 CP8EH9 46885653 IC50 = 13.7 nM T85467 C23VOP 46885654 IC50 = 15 nM T85467 C1D7HM 46885655 IC50 = 1.6 nM T85467 C6GU4W 46885656 IC50 = 1 nM T85467 CGR48P 46885686 IC50 = 3.2 nM T85467 CKNF58 46885687 IC50 = 0.6 nM T85467 C5G0CV 46885688 IC50 = 0.3 nM T85467 CQ48VM 46885689 IC50 = 0.6 nM T85467 C2FR7X 46885690 IC50 = 0.9 nM T85467 CN8D5V 46885691 IC50 = 1.6 nM T85467 C9WME2 46885732 IC50 = 2.8 nM T85467 CAZ2X9 46885733 IC50 = 0.6 nM T85467 CC5IS8 46885734 IC50 = 0.9 nM T85467 C9RP0X 46885735 IC50 = 0.6 nM T85467 CWV65J 46885783 IC50 = 39 nM T85467 C6C2DF 46885784 IC50 = 64 nM T85467 CAXI18 46885785 IC50 = 237 nM T85467 CG4L0I 46885786 IC50 = 0.2 nM T85467 CFI0D2 46885837 IC50 = 0.2 nM T85467 CNU9K2 46885838 IC50 = 5.5 nM T85467 CME71U 46885839 IC50 = 0.2 nM T85467 C2FJ9M 46885840 IC50 = 1.1 nM T85467 CRPW37 46885881 IC50 = 0.2 nM T85467 CGX8P2 46885882 IC50 = 11.6 nM T85467 C8J3XO 46885883 IC50 = 201.8 nM T85467 C6J7KC 46885945 IC50 = 0.3 nM T85467 C45SRZ 46885946 IC50 = 0.2 nM T85467 C5JEH0 46885947 IC50 = 4.5 nM T85467 C2EC9H 46885984 IC50 = 1.9 nM T85467 C8IUJ6 46885985 IC50 = 2.7 nM T85467 CYV9C4 46885986 IC50 = 125.1 nM T85467 C9TCR1 46886026 IC50 = 7.2 nM T85467 C63CFU 46886027 IC50 = 16.5 nM T85467 C2GZ0M 46886028 IC50 = 1.3 nM T85467 C8DU2J 46886029 IC50 = 1.3 nM T85467 C0A2CI 46890616 Ki >= 504 nM T85467 CW52VH 46890658 Ki >= 260 nM T85467 CXQ2W0 46890659 Ki >= 580 nM T85467 CQ20RC 46890660 Ki >= 100 nM T85467 CTR7Q0 49850345 Ki = 5.012 nM T85467 C0ZOG4 49850346 Ki = 3.162 nM T85467 CW7H3I 49850347 Ki = 6.31 nM T85467 C38XUQ 49850348 Ki = 19.95 nM T85467 CM06FG 50898361 Ki = 530 nM T85467 C4Q9NK 50899741 Ki = 6.31 nM T85467 CU78LF 52940662 Ki = 1258.93 nM T85467 C9VIG1 52940697 Ki = 2511.89 nM T85467 CS5MB6 52940700 Ki = 1258.93 nM T85467 C1NI2M 52940701 Ki > 25118.86 nM T85467 COZ3W6 52940918 Ki > 25118.86 nM T85467 C4H2AR 52941063 Ki = 1000 nM T85467 CBV71O 52941863 Ki = 1258.93 nM T85467 CY7WR1 52941873 Ki = 794.33 nM T85467 CK73QL 52941886 Ki = 1995.26 nM T85467 C9ZHY5 52941891 Ki = 1258.93 nM T85467 CKGU98 52943098 Ki = 5011.87 nM T85467 C8KGO6 52943112 Ki > 25118.86 nM T85467 C1UV3M 52943117 Ki = 125.89 nM T85467 CF8X6C 52943118 Ki = 199.53 nM T85467 C2EM1L 52944267 Ki > 25118.86 nM T85467 C4YZS8 52944290 Ki = 100 nM T85467 C40PIO 52944303 Ki > 25118.86 nM T85467 C81GXN 52944309 Ki = 158.49 nM T85467 C4KL9X 52944419 Ki > 25118.86 nM T85467 CLHD03 52944708 Ki = 398.11 nM T85467 CF1ZU9 52945294 Ki = 8 nM T85467 CLJO68 52945504 Ki = 398.11 nM T85467 CXY80T 52945505 Ki = 501.19 nM T85467 CBF7V9 52946459 Ki = 794.33 nM T85467 CPWL93 52946711 Ki = 501.19 nM T85467 CFI4T3 52946739 Ki = 125.89 nM T85467 CX49CM 52946740 Ki = 125.89 nM T85467 CH6C7Q 52946754 Ki = 199.53 nM T85467 C62ANP 52946882 Ki = 251.19 nM T85467 C4K6BH 52946883 Ki = 50.12 nM T85467 CF9XJ7 52946975 Ki > 25118.86 nM T85467 C5V9JN 52947148 Ki = 1000 nM T85467 CR1V4J 52947169 Ki > 25118.86 nM T85467 C4PF1S 52947722 Ki = 63.1 nM T85467 CP7UZ9 52947935 Ki = 3162.28 nM T85467 CB59YF 52947936 Ki > 25118.86 nM T85467 CJK63Q 52948954 Ki = 3981.07 nM T85467 C26JAX 52948962 Ki = 1000 nM T85467 C47ORF 52949154 Ki > 25118.86 nM T85467 C8OV5R 52949166 Ki = 398.11 nM T85467 CYMR14 52949167 Ki > 25118.86 nM T85467 C9OWA1 52949168 Ki > 25118.86 nM T85467 C0HA6F 52949188 Ki = 25.12 nM T85467 C1P3MV 52949428 Ki > 25118.86 nM T85467 C3H1YG 52950153 Ki = 1584.89 nM T85467 C0SU2P 53234014 Ki = 6.31 nM T85467 CC4YD0 54580770 Ki = 316.23 nM T85467 CEKY15 54580771 Ki = 3162.28 nM T85467 CIO2K9 54581783 Ki = 50.12 nM T85467 CPN3U5 54581784 Ki = 7.943 nM T85467 C6CI7U 54581785 Ki = 39.81 nM T85467 CB81XY 54581786 Ki = 19.95 nM T85467 C5JEO4 54582745 Ki = 15.85 nM T85467 C6AYV4 54582746 Ki = 199.53 nM T85467 CMFT46 54582747 Ki > 25118.86 nM T85467 CY5C7W 54582748 Ki = 50.12 nM T85467 CU87RC 54583735 Ki = 31.62 nM T85467 CSHM03 54583736 Ki = 1584.89 nM T85467 CKGL87 54583737 Ki = 39.81 nM T85467 CA5VR8 54583738 Ki = 1258.93 nM T85467 CN6PE1 54583739 Ki = 794.33 nM T85467 C4SG0X 54584713 Ki = 7.943 nM T85467 CN7B1S 54584714 Ki = 501.19 nM T85467 C2HQ1E 54584715 Ki > 25118.86 nM T85467 CJL52D 54586642 Ki = 125.89 nM T85467 C75KAS 54586643 Ki = 79.43 nM T85467 CQV1T2 54586644 Ki = 7.943 nM T85467 C8OY2R 54587664 Ki = 19.95 nM T85467 C0X1JB 54587665 Ki = 2511.89 nM T85467 C4YHT2 54587666 Ki = 630.96 nM T85467 CWR1Z7 56665984 Ki > 13000 nM T85467 C96FQZ 57395059 EC50 = 3000 nM T85467 CP7A2U 58905349 IC50 > 20000 nM T85467 CB1N8J 58905358 IC50 > 20000 nM T85467 C1CFM4 58905388 IC50 > 20000 nM T85467 C0U1HA 59179260 Ki > 5000 nM T85467 CK7T6D 59179887 Ki > 5000 nM T85467 C4CIH9 59179917 Ki > 5000 nM T85467 CVC72I 59554822 EC50 = 3.9 nM T85467 CCXA68 59554824 EC50 = 50 nM T85467 C2EVC3 59554827 EC50 = 8.4 nM T85467 CNUA34 66857670 EC50 = 18 nM T85467 C1WA3L 66857738 EC50 = 6.7 nM T85467 C1C3AF 66857975 EC50 = 8.8 nM T85467 CUIV04 66857988 EC50 = 3.3 nM T85467 CB56OD 66858036 EC50 = 36 nM T85467 CU5V8I 66858111 EC50 = 27 nM T85467 CB2J4V 66978356 EC50 = 0.91 nM T85467 C4FHO2 67082722 EC50 = 16 nM T85467 CGQA79 67082748 EC50 = 3.5 nM T85467 CVM9Q1 68503758 IC50 > 25000 nM T85467 CA15ND 68505312 IC50 > 25000 nM T85467 C0US2T 68505327 IC50 > 25000 nM T85467 CX8W7F 68508048 IC50 > 25000 nM T85467 CI0A9L 68747456 EC50 = 2700 nM T85467 C6IHR3 68747472 EC50 = 4700 nM T85467 C5NZO0 68747479 EC50 = 4 nM T85467 C8MED0 68749474 EC50 = 18 nM T85467 CIUR89 68751402 EC50 = 13 nM T85467 C8WC4E 68785185 EC50 = 27 nM T85467 CJ7AY6 69753740 EC50 = 3.6 nM T85467 CITN25 71451558 Ki = 678.4 nM T85467 C01YOJ 71452690 Ki = 1000 nM T85467 CQ5E0J 71455094 Ki = 26 nM T85467 CY17WU 71456904 Ki = 218.5 nM T85467 C81JRT 71458756 Ki = 23.4 nM T85467 COK0V6 71458757 Ki = 135 nM T85467 CWU68H 71460570 Ki = 1496.8 nM T85467 CJRI61 71461205 Ki = 9.9 nM T85467 C74PUE 71462285 Ki = 18 nM T85467 CS5U2J 71462286 Ki = 1264.6 nM T85467 C8XJ0I 71733818 IC50 > 25000 nM T85467 CXC78L 71733909 IC50 > 25000 nM T85467 C7B5XE 71733910 IC50 > 25000 nM T85467 CQ21ZD 71733911 IC50 > 25000 nM T85467 CZG0S2 71733912 IC50 > 25000 nM T85467 C4G2UR 72695027 Ki > 12700 nM T85467 CDFO42 72695136 Ki > 14000 nM T85467 CX6T7A 72706947 Ki = 880 nM T85467 C6PLC5 72722131 Ki = 258 nM T85467 CU39ZO 72950089 Ki = 350 nM T85467 C4T8HI 91668213 Ki = 2 nM T85467 CWTO83 91810751 Ki > 14000 nM T85467 C1LWP5 91827668 Ki = 11.7 nM T85467 C2QJ3O 117993349 Ki = 31.6 nM T85467 CR64HV 117993400 Ki = 3.6 nM T85467 CQK9R7 117993413 Ki = 7.8 nM T85467 CR4DE7 118175009 Ki > 17500 nM T85467 CSJ4A9 118352160 EC50 > 10000 nM T85467 CE6L8I 118352177 EC50 > 10000 nM T85467 C8PKA7 118352211 EC50 > 10000 nM T85467 CPS7M4 118352285 EC50 > 10000 nM T85467 C7Z3HU 122180289 IC50 > 30000 nM T85467 C2NG1J 122180295 IC50 > 30000 nM T85467 C8ZRJ0 126495398 EC50 = 5800 nM T85467 C8SRZ5 126495427 EC50 > 10000 nM T85467 CD72CT 126495432 EC50 > 10000 nM T85467 CN72WL 126495463 EC50 = 1400 nM T85467 CV1A6C 126495491 EC50 = 360 nM T85467 CYP3E5 126495507 EC50 > 10000 nM T85467 C2N7XJ 127026652 EC50 = 2606 nM T85467 CX9M6D 127029402 EC50 > 10000 nM T85467 CWXR72 127029417 Ki > 50000 nM T85467 CW1O4F 127029692 EC50 > 10000 nM T85467 C0UJ5N 127037150 EC50 = 310 nM T85467 C94QAU 127046040 Ki = 64.5 nM T85467 C94NDQ 127046263 Ki = 14.5 nM T85467 CIY0C1 127046264 Ki = 16.5 nM T85467 C01ACX 127046441 Ki = 10 nM T85467 CX6DG8 127047210 Ki = 53.1 nM T85467 CJAQ90 127047381 Ki > 50000 nM T85467 CBCQ64 127047601 IC50 = 74.3 nM T85467 CI6G4K 127047602 Ki = 1066 nM T85467 C7OHJ8 127047603 Ki = 5890 nM T85467 C2KU5J 127047604 Ki = 310 nM T85467 CU78GX 127047605 Ki = 584 nM T85467 CH78WV 127047606 Ki > 9650 nM T85467 CX39ZL 127047729 Ki = 14.1 nM T85467 C59JLB 127048124 Ki = 38.3 nM T85467 CTR62O 127052613 EC50 = 0.8 nM T85467 CGZR45 127052614 EC50 = 260 nM T85467 COVY75 127052615 EC50 = 7600 nM T85467 C4U3XA 134138103 EC50 = 540 nM T85467 C10OQL 134144861 EC50 = 6400 nM T85467 CG0SO1 134147356 EC50 = 2.3 nM T85467 C8QT5L 134149776 EC50 = 4800 nM T85467 C16HYX 134151657 EC50 = 130 nM T85467 CIA76T 134157766 EC50 = 870 nM T85467 CA8QC3 141730897 IC50 = 2292.3 nM T85467 C2P9GV 141730900 IC50 > 10000 nM T85467 CK6E7L 141730914 IC50 > 10000 nM T85467 C7B5WG 141730916 IC50 > 10000 nM T85467 C62DUY 141730923 IC50 > 10000 nM T85467 CSXG54 145965248 EC50 = 3.4 nM T85467 CIS1V8 145966519 EC50 = 32 nM T85467 C54SAN 145971909 EC50 = 0.8 nM T85467 CGV2E8 145977227 EC50 = 1 nM T85467 CLVI73 145978309 EC50 = 3 nM T85467 CDN70S 146014480 IC50 > 10000 nM T85467 CZ10RG 155522808 IC50 > 10000 nM T85467 C7UY3Q 155529786 IC50 > 10000 nM T85467 C82RVN 155554217 IC50 > 10000 nM T85467 D02LXJ 9813912 Ki = 100 nM T85467 D02MXT 24952929 Ki > 7900 nM T85467 D02SAD 44419388 Ki = 68 nM T85467 D03OYD 5311240 IC50 = 3100 nM T85467 D05TNX 5311100 EC50 = 3400 nM T85467 D07JMB 44289922 Ki = 1175 nM T85467 D07UDT 15551229 Ki = 0.6 nM T85467 D08MNO 25886893 Ki > 10000 nM T85467 D08ZYC 11595431 Ki = 398.11 nM T85467 D0H5TU 11524454 IC50 > 20000 nM T85467 D0J9PG 119461 Ki = 1600 nM T85467 D0O9ES 5311053 IC50 = 635 nM T85467 D0S2LO 9864831 Ki > 13000 nM T85467 D0TA0L 23685469 Ki > 1000 nM T85467 D0Y1IF 23664784 Ki > 10000 nM T85467 D0Z3XJ 9817405 Ki = 20 nM T70521 CLW69A 656970 Ki = 0.002 nM T70521 CW4CT3 2091305 Ki = 17000 nM T70521 CH5X4Y 2777630 Ki = 5200 nM T70521 C7DT0M 3006281 Ki = 20 nM T70521 CWQ43C 3006282 Ki = 100 nM T70521 C8FG3C 3006283 Ki = 36 nM T70521 CXAD51 3006284 Ki = 1.6 nM T70521 CHZX14 3006285 Ki = 3.4 nM T70521 CGY39U 3006286 Ki = 3.9 nM T70521 CO6D8V 3006287 Ki = 8.1 nM T70521 C6NV0O 3011183 Ki = 2800 nM T70521 C4AO1T 3011184 Ki = 1000 nM T70521 C4XV5O 3011185 Ki = 22000 nM T70521 CK8P0G 3011186 Ki = 64000 nM T70521 CP3A5D 3011187 Ki = 27000 nM T70521 C7TMP4 3011188 Ki = 4000 nM T70521 CU5PZ6 3011189 Ki = 11000 nM T70521 C0BE1Q 3011190 Ki = 760 nM T70521 C81QKX 3011191 Ki = 500 nM T70521 C07AIZ 3011192 Ki = 1200 nM T70521 CNL9Y1 3011193 Ki = 2700 nM T70521 C0BJQ8 3011194 Ki = 4900 nM T70521 C5AL7S 3011195 Ki = 6500 nM T70521 COQ27C 3011196 Ki = 2200 nM T70521 C2W8RM 3011197 Ki = 1800 nM T70521 CIG57B 3011198 Ki = 2300 nM T70521 C62KAT 3011199 Ki = 12.5 nM T70521 C35DET 3011200 Ki = 28.5 nM T70521 CHO6W7 3011201 Ki = 52 nM T70521 CW6J0E 3011202 Ki = 11 nM T70521 CPQ9N1 3011203 Ki = 14.6 nM T70521 CM72DB 3011204 Ki = 13 nM T70521 C3PCR7 3011205 Ki = 17 nM T70521 C4X9QK 3011206 Ki = 36 nM T70521 C41JZM 3011207 Ki = 94 nM T70521 C7T1XL 3011208 Ki = 25 nM T70521 CCV10J 3011209 Ki = 191 nM T70521 CG3W1Z 3011210 Ki = 240 nM T70521 CR0H4V 3011211 Ki = 498 nM T70521 C29WHE 3011212 Ki = 125 nM T70521 C3FB9J 5270924 Ki = 10.8 nM T70521 CP2Z5T 11653830 Ki = 1.7 nM T70521 C90ICD 24799124 Ki = 0.84 nM T70521 C63YXN 24799125 Ki = 0.45 nM T97149 D05ADP 160355 IC50 > 10000 nM T97149 D0E3TC 44259 IC50 = 34.8 nM T97149 D00OWF 5280953 IC50 = 410 nM T97149 D0NS6I 10037501 IC50 = 1400 nM T97149 D0PO8N 117881270 IC50 = 99 nM T97149 D0Q3VZ 135398522 IC50 = 320 nM T97149 CVMO57 95875 IC50 > 10000 nM T97149 CQ0ZI7 45141513 IC50 = 16000 nM T97149 CDK93W 56946894 IC50 = 40 nM T97149 CR3I5F 57418686 IC50 = 3000 nM T97149 CF6K1Y 58857683 IC50 = 15000 nM T97149 C56MAG 59379853 IC50 > 10000 nM T97149 CV63UL 67240318 IC50 > 10000 nM T97149 CF7R0Y 71682057 IC50 = 10000 nM T97149 CVD5U4 76314850 IC50 = 2200 nM T97149 C0GYK1 86765296 IC50 = 1200 nM T97149 C4BKA6 89429109 IC50 > 10000 nM T97149 C2FOK4 89494280 IC50 = 1700 nM T97149 CE5L8V 90388565 IC50 = 4700 nM T97149 CWE9I2 91664021 IC50 > 10000 nM T97149 CW58AE 91664022 IC50 > 10000 nM T97149 CB25UZ 91664023 IC50 > 10000 nM T97149 CO83PN 122181013 IC50 > 100000 nM T97149 C69ULZ 122181014 IC50 > 100000 nM T97149 CIG8Y1 122181016 IC50 = 2300 nM T97149 CRJS41 122181017 IC50 > 10000 nM T97149 CVB03H 122181018 IC50 = 1400 nM T97149 C6SJ3X 122181019 IC50 > 10000 nM T97149 C7L5PG 122181021 IC50 > 10000 nM T97149 C58CJI 122181022 IC50 > 10000 nM T97149 CC2G8N 122181024 IC50 = 30 nM T97149 CV5BQ9 122181097 IC50 > 10000 nM T97149 C2LWZ1 129318964 IC50 > 10000 nM T97149 C4Q5LF 132471857 IC50 = 54 nM T97149 CM8DK3 134813913 IC50 = 380 nM T97149 CBU0J4 135604653 IC50 > 10000 nM T97149 CH0Q2Z 136234577 IC50 = 200 nM T97149 CV6F4N 136234578 IC50 = 180 nM T97149 C2G3JY 136234579 IC50 > 10000 nM T97149 CCAZ26 137631656 IC50 = 920 nM T97149 C3QAV9 137631819 IC50 = 3000 nM T97149 CG8Y0U 137633419 IC50 = 17000 nM T97149 CS9TU2 137633985 IC50 = 7900 nM T97149 C83UKG 137634382 IC50 = 120 nM T97149 CNT7S3 137634818 IC50 > 10000 nM T97149 CCP7X5 137635304 IC50 = 4900 nM T97149 C1AK8X 137635556 IC50 = 1100 nM T97149 CV7OF5 137635713 IC50 > 10000 nM T97149 C5QWE1 137635926 IC50 = 110 nM T97149 CKZF46 137638065 IC50 > 10000 nM T97149 CCX37E 137638472 IC50 = 2100 nM T97149 CPO87L 137638509 IC50 = 110 nM T97149 C1UI5N 137638944 IC50 = 8100 nM T97149 CH4RP3 137639514 IC50 = 430 nM T97149 CX3MQ1 137639546 IC50 = 1400 nM T97149 CH3S8N 137640038 IC50 = 140 nM T97149 CXM4G7 137640811 IC50 = 320 nM T97149 CF83TG 137640934 IC50 = 5300 nM T97149 CWVE69 137643514 IC50 = 1200 nM T97149 CYA1F7 137643721 IC50 = 1300 nM T97149 C2AG3W 137643887 IC50 = 41000 nM T97149 C4DS3I 137643955 IC50 = 5100 nM T97149 CWIP72 137644498 IC50 = 1800 nM T97149 CZ4U0W 137644802 IC50 > 100000 nM T97149 CPJ42V 137644974 IC50 > 10000 nM T97149 C8VTQ9 137645650 IC50 = 320 nM T97149 C7ZOV3 137645947 IC50 > 10000 nM T97149 CL5NX9 137646497 IC50 = 610 nM T97149 CJ5O2Q 137646673 IC50 > 10000 nM T97149 COU37W 137647335 IC50 = 3100 nM T97149 C7O2AW 137647969 IC50 > 10000 nM T97149 C5OJH2 137649318 IC50 = 510 nM T97149 C9QNG8 137650421 IC50 = 10000 nM T97149 CWG94C 137650926 IC50 = 10000 nM T97149 C8MKN0 137651314 IC50 = 910 nM T97149 CKL0P4 137651538 IC50 = 3900 nM T97149 CJ14XO 137651668 IC50 = 2300 nM T97149 CH6L2T 137652047 IC50 = 7100 nM T97149 C2B5CY 137652970 IC50 = 6600 nM T97149 C48DVU 137653000 IC50 = 930 nM T97149 C01URE 137653446 IC50 > 10000 nM T97149 C47FBV 137654225 IC50 = 1900 nM T97149 C7IU4J 137655848 IC50 = 460 nM T97149 CQEJ60 137656868 IC50 = 520 nM T97149 C39SEV 137658150 IC50 = 2100 nM T97149 CX8YL9 137658187 IC50 = 81 nM T97149 CA2PY1 137658970 IC50 = 1700 nM T97149 CJ1TB2 137659239 IC50 > 10000 nM T97149 C3U2OB 137659350 IC50 = 950 nM T97149 C7MI2G 137661183 IC50 > 10000 nM T97149 CIX41F 137661315 IC50 > 10000 nM T97149 CD0FV8 137661355 IC50 = 5300 nM T97149 CZ9BN4 138320062 IC50 = 0.104 nM T97149 C2MD1Q 155513187 IC50 > 10000 nM T97149 D00ERW 44444843 Ki > 5804 nM T97149 D04TPA 72163809 IC50 = 70 nM T97149 D0A7FQ 11644425 IC50 = 3200 nM T59493 CW9SF3 81732 IC50 = 1200000 nM T59493 CV7T4F 71656047 IC50 = 3700 nM T59493 CB54NU 122177329 IC50 = 664000 nM T59493 C3H2AM 122177330 IC50 = 436000 nM T59493 CT8WJ6 122177331 IC50 = 312000 nM T59493 CYVR40 122177338 IC50 = 776000 nM T59493 C7K5MP 122177342 IC50 = 832000 nM T59493 CRG32Y 122177345 IC50 = 677000 nM T59493 CKT52Z 122177346 IC50 = 697000 nM T59493 CVA04H 122177347 IC50 = 30000 nM T59493 C8RX9F 127026008 IC50 = 48300 nM T59493 CV7WK1 127026009 IC50 = 69100 nM T59493 C2QW4P 127026010 IC50 = 17600 nM T59493 CEAV32 127035811 IC50 = 11900 nM T59493 CTK1M4 127035812 IC50 = 26000 nM T59493 CP8KT1 127035813 IC50 = 33800 nM T59493 CM8AT2 127035814 IC50 = 11500 nM T59493 C4NOX1 127035846 IC50 = 59600 nM T59493 CFV98O 127035847 IC50 = 7200 nM T59493 CBE69J 127035848 IC50 = 40100 nM T59493 CKZ15S 127035849 IC50 = 50800 nM T59493 C7JV5R 127035870 IC50 = 25600 nM T59493 CU7Y5G 127035871 IC50 = 9600 nM T59493 C9A8TW 127035872 IC50 = 17500 nM T59493 C3VH6Q 127035985 IC50 = 33700 nM T59493 CMQ6P8 127036013 IC50 = 7900 nM T59493 CQ68CM 127036014 IC50 = 13700 nM T59493 C0RT2Y 127036648 IC50 = 141700 nM T59493 CCEB19 127037439 IC50 = 57200 nM T53024 D02XIY 448601 Ki = 0.4 nM T53024 D0TV0C 9941444 Ki = 1 nM T53024 D06JFI 11251755 IC50 = 41 nM T53024 D0J8PI 158782 IC50 = 14 nM T53024 D09JXL 5311430 Ki = 0.07943 nM T53024 D0Y2HR 2247 Ki > 10000 nM T53024 C6XYL5 6918011 Ki = 0.5012 nM T53024 CHM63P 6918026 Ki = 0.07943 nM T53024 CR0U6E 9827283 Ki = 46 nM T53024 CA8UQ7 9848232 Ki = 615 nM T53024 CW3TM5 9851998 Ki = 0.5 nM T53024 CTRI07 9852911 Ki = 1800 nM T53024 C9BJ3Q 9854636 IC50 = 807 nM T53024 CS2D0V 9872511 Ki = 2500 nM T53024 C71BKL 9893924 Ki = 621 nM T53024 CMLP16 9918828 Ki = 0.631 nM T53024 CRP01W 9959684 Ki = 1000 nM T53024 CF6TA4 9959983 IC50 = 0.2 nM T53024 C3Z5YJ 9963342 Ki = 1.995 nM T53024 CIT57N 9985523 Ki = 3100 nM T53024 C64LIB 10009650 Ki = 800 nM T53024 C58EOI 10053855 Ki = 2.1 nM T53024 C0NQ9G 10054314 IC50 = 0.2 nM T53024 CL6G0Z 10094509 Ki = 6180 nM T53024 C9C7RK 10096510 Ki = 9500 nM T53024 CFZN71 10166743 Ki = 3470 nM T53024 CI21CK 10179247 Ki > 10000 nM T53024 C6DRE9 10210016 Ki > 10000 nM T53024 C4M9GN 10248767 Ki = 7900 nM T53024 CSY5K2 10325243 Ki = 4600 nM T53024 C67NLY 10369961 Ki = 778 nM T53024 CL87OB 10411795 Ki > 10000 nM T53024 CP2S9D 10436888 Ki = 4200 nM T53024 C0YFD4 10505242 Ki = 2300 nM T53024 CN3IV5 10528970 Ki = 33000 nM T53024 CJ40IE 10531093 Ki = 565 nM T53024 CS96ON 10534086 IC50 = 183 nM T53024 CRZ9I3 10553122 Ki = 8000 nM T53024 CB2NK4 10554498 Ki = 310 nM T53024 CA1VI4 10554709 Ki = 3000 nM T53024 CHZ9I8 10554930 Ki = 4600 nM T53024 CY3ZE9 10577746 IC50 = 1585 nM T53024 CIY02U 10578474 Ki = 1700 nM T53024 C9C0HF 10580397 Ki = 600 nM T53024 CUW4E5 10601454 Ki = 1000 nM T53024 CD8ZW7 10602230 Ki = 894 nM T53024 C1M5RT 10602592 Ki = 53 nM T53024 CVY6D0 10603005 Ki > 300000 nM T53024 CD4HA5 10624774 Ki = 300 nM T53024 CGZ6W8 10625454 Ki = 500 nM T53024 C0SXF1 10625762 Ki = 830 nM T53024 CU3DQ6 10630127 Ki = 5.51 nM T53024 C15AHJ 10650427 Ki = 2200 nM T53024 C7AX8J 10650940 Ki = 777 nM T53024 C5UOS4 10698494 Ki > 300000 nM T53024 CT81RB 10698706 Ki > 300000 nM T53024 C45JIZ 10699714 Ki = 2700 nM T53024 CG2UX4 10701257 IC50 = 291 nM T53024 C27FVZ 10720221 Ki = 12000 nM T53024 CP0F7C 10724811 IC50 = 1000 nM T53024 C3TMY5 10724880 IC50 = 306 nM T53024 CK7R2B 10745635 Ki = 2000 nM T53024 CJM47E 10748701 IC50 = 118 nM T53024 CWF2N5 10748831 IC50 = 82.5 nM T53024 CLQ07H 10768264 Ki = 2000 nM T53024 C4X2CO 10769191 Ki = 1600 nM T53024 CLW4V6 10770814 Ki = 2600 nM T53024 CO56HI 10772403 IC50 = 566 nM T53024 CGN0Z5 10772578 IC50 = 123 nM T53024 COY17C 10793795 Ki > 300000 nM T53024 C3L4DH 10796238 IC50 = 350 nM T53024 C0WND2 10815650 Ki = 114000 nM T53024 C61EOJ 10816544 Ki = 74000 nM T53024 C15QGO 10819673 IC50 = 1000 nM T53024 CFU8M6 10838621 Ki = 10000 nM T53024 CJ4T3I 10841338 Ki = 1700 nM T53024 CFL71O 10843862 IC50 = 445 nM T53024 C2PJ1O 10876898 Ki = 3.162 nM T53024 C6TVQ8 10964197 Ki = 10 nM T53024 CXDG12 10996788 Ki = 0.5012 nM T53024 C6AW0M 11112736 Ki > 10000 nM T53024 CK1RX4 11136828 Ki = 0.7943 nM T53024 CR1JP9 11147505 Ki = 0.7943 nM T53024 C1I9EX 11159133 IC50 > 1000 nM T53024 C7REL4 11170698 IC50 = 25.7 nM T53024 CIEM12 11170867 IC50 = 1.5 nM T53024 CW2JA8 11182381 IC50 = 30 nM T53024 CE3GC2 11205475 IC50 = 130 nM T53024 CXI32T 11205496 IC50 = 71 nM T53024 C2RNJ5 11205515 IC50 = 170 nM T53024 CUT8Z0 11240205 IC50 = 27 nM T53024 CK78SD 11240206 IC50 = 54 nM T53024 C67WXD 11274767 IC50 = 15.5 nM T53024 COK06N 11320738 IC50 = 194 nM T53024 C5D6AM 11332138 IC50 = 183 nM T53024 C5PAN4 11343811 IC50 = 227 nM T53024 CLQ53A 11355270 IC50 = 30 nM T53024 CQ0UC7 11378229 IC50 = 173 nM T53024 CC09ZU 11378299 IC50 = 622 nM T53024 CG7PT9 11389178 IC50 > 1000 nM T53024 CFJD72 11423410 IC50 = 57 nM T53024 C4S2HG 11434734 IC50 = 40 nM T53024 C3T6XG 11442741 Ki > 5000 nM T53024 C6XHC3 11457491 IC50 = 347 nM T53024 CJ5A9B 11457521 IC50 = 120 nM T53024 CMA8C7 11468709 IC50 > 1000 nM T53024 CG8A0J 11468887 IC50 = 43 nM T53024 CZ3N5J 11468916 IC50 = 52 nM T53024 CORY59 11480246 IC50 = 12 nM T53024 C63QMX 11535351 IC50 = 49 nM T53024 CF6K7M 11563877 IC50 = 0.17 nM T53024 CP4DH2 11614416 IC50 = 0.53 nM T53024 CS68YA 11642413 IC50 = 980 nM T53024 CZHN61 11678313 IC50 > 10000 nM T53024 CW65KY 11705763 Ki = 2 nM T53024 CN63YV 11787877 IC50 = 962 nM T53024 CR6UF9 11788180 IC50 > 1000 nM T53024 CK7BN1 11800917 Ki = 2000 nM T53024 CK4U8N 11804376 IC50 = 797 nM T53024 C9XH7F 11815114 Ki = 0.7943 nM T53024 CUI15C 11828523 IC50 = 2250 nM T53024 CRA01O 11845058 IC50 = 6.2 nM T53024 C8X3CL 11845059 IC50 = 3.1 nM T53024 CO3HT9 11847587 IC50 = 7.5 nM T53024 CAD8P9 11848624 Ki > 10000 nM T53024 CM49QW 11848625 Ki > 10000 nM T53024 CEBA46 11848626 Ki > 10000 nM T53024 CCT5G7 11848677 Ki > 10000 nM T53024 CMR10F 11848679 Ki > 10000 nM T53024 C9QDX3 11848833 Ki > 10000 nM T53024 CL6B5X 11848835 Ki > 10000 nM T53024 CBV2X0 11963995 Ki > 10000 nM T53024 CW7I8U 13690207 IC50 = 0.02 nM T53024 C8OU7I 15429504 IC50 = 34.8 nM T53024 CEO3F0 15585102 IC50 = 18 nM T53024 CC2YJ8 16062553 Ki > 10000 nM T53024 C3H1RT 16062555 Ki > 10000 nM T53024 C1LH5T 16062816 Ki > 10000 nM T53024 C1GKF8 16130982 Ki = 0.001 nM T53024 C41XOQ 16133849 EC50 = 2.3 nM T53024 C2TRA5 16144717 IC50 = 202 nM T53024 CW20OC 16144977 IC50 = 75.9 nM T53024 CS6A3Z 16145268 IC50 = 46.1 nM T53024 CN3LS1 16145579 IC50 = 144 nM T53024 C72MUC 16146425 IC50 = 68.5 nM T53024 CD91IL 16148220 IC50 = 706 nM T53024 C59OUC 16148481 Ki = 19.95 nM T53024 CJG1X9 16148596 Ki = 6.31 nM T53024 CNY09C 16148922 Ki = 1000 nM T53024 CP0DC8 16149640 Ki = 1.259 nM T53024 CDPC19 16149975 Ki = 1 nM T53024 C0SE6V 16150676 Ki = 0.1259 nM T53024 CSP6A9 16150915 Ki = 0.07943 nM T53024 C6N7SR 16151159 Ki = 19.95 nM T53024 C2B9IL 16151570 IC50 > 1000 nM T53024 CQM8J1 16151781 IC50 = 550 nM T53024 CM8UF7 16151826 IC50 > 1000 nM T53024 CJ7UT6 16151923 IC50 > 1000 nM T53024 CIM03U 16152257 IC50 = 260 nM T53024 CU7X6V 16153077 IC50 = 48 nM T53024 CK4O1V 16153193 IC50 = 56 nM T53024 C16LMW 16153418 IC50 = 700 nM T53024 CO0LG7 16154000 IC50 = 561 nM T53024 CX4RM8 16154096 IC50 = 179 nM T53024 COYU86 16156815 Ki = 1000 nM T53024 CI3FW1 16157160 IC50 = 48.2 nM T53024 C7GN0S 16157479 Ki = 0.1585 nM T53024 CQL5O0 16181427 IC50 > 1000 nM T53024 C2CUY9 16181428 IC50 > 1000 nM T53024 CUH8D7 16737812 IC50 = 357 nM T53024 C8QIT3 16737813 IC50 > 1000 nM T53024 CNP36U 16737814 IC50 = 83 nM T53024 C7Q6JL 16738359 IC50 = 103 nM T53024 CJ9K1C 24740750 Ki > 10000 nM T53024 CS6VO9 24740751 Ki > 10000 nM T53024 CA4K0B 24740752 Ki > 10000 nM T53024 C4N3AX 24740753 Ki > 10000 nM T53024 COQU12 24740861 Ki > 10000 nM T53024 CAD4S1 24740862 Ki > 10000 nM T53024 C67YVI 24740863 Ki > 10000 nM T53024 CO0IF5 24740864 Ki > 10000 nM T53024 C6F1RZ 24777672 IC50 > 1000 nM T53024 C5GZO7 24858018 IC50 = 6.5 nM T53024 CV1U7H 24858920 IC50 = 14.5 nM T53024 C0UB7K 24859055 IC50 = 11 nM T53024 CQCW58 24859056 IC50 = 49 nM T53024 CT6J2A 24859195 IC50 = 8 nM T53024 CUDV69 24859196 IC50 = 4.9 nM T53024 C45NYA 24859341 IC50 = 9 nM T53024 C4AB6I 24859342 IC50 = 42 nM T53024 CH50QU 24859494 IC50 = 33 nM T53024 C8L2KJ 24859495 IC50 = 5.4 nM T53024 CDS6W5 24859645 IC50 = 41 nM T53024 CHF20D 24859646 IC50 = 4.8 nM T53024 CKH2R4 24859787 IC50 = 18.5 nM T53024 CT1BM6 24859788 IC50 = 13 nM T53024 C2IKX3 24859919 IC50 = 11 nM T53024 C5OQ2X 24859920 IC50 = 109 nM T53024 CSZ73L 24860057 IC50 = 3.9 nM T53024 C36ZHQ 24860058 IC50 = 13 nM T53024 CVL48C 24860201 IC50 = 34 nM T53024 C20ZFS 24860202 IC50 = 40 nM T53024 CL20IX 24951595 Ki = 1.5 nM T53024 CMOV54 24951597 Ki = 0.038 nM T53024 CJO4V0 24951598 Ki = 0.037 nM T53024 CWY8N5 24952323 Ki = 0.08 nM T53024 CZJ6P0 24952682 Ki = 0.1 nM T53024 COH85D 24953027 Ki = 0.11 nM T53024 C49PIW 24953029 Ki = 0.12 nM T53024 CM12PG 24956953 Ki = 0.08 nM T53024 CHKC79 25187396 IC50 = 292 nM T53024 C4YXJ1 25187398 IC50 = 10 nM T53024 CO9PI7 25187400 IC50 = 103 nM T53024 C8C9PL 25187679 IC50 = 22 nM T53024 C9ECD8 25187681 IC50 = 12 nM T53024 C43OES 25187683 IC50 = 242 nM T53024 CNTB73 25187685 IC50 = 2.1 nM T53024 C1IUQ2 25187953 IC50 = 327 nM T53024 CQ3F8L 25187955 IC50 = 2.1 nM T53024 CS2ZV1 25188218 IC50 = 770 nM T53024 CLI2U1 25188220 IC50 = 452 nM T53024 CNDU95 25188496 IC50 = 290 nM T53024 C7KF8N 25188776 IC50 > 1000 nM T53024 CCHN50 25188780 IC50 > 1000 nM T53024 C3T8DA 25189052 IC50 = 0.73 nM T53024 CI21ED 25189054 IC50 = 4.2 nM T53024 C97LHK 25189325 IC50 = 183 nM T53024 CEG4J0 25189327 IC50 = 215 nM T53024 CSQH26 42637069 IC50 > 1000 nM T53024 CJ1S9K 42637136 IC50 > 1000 nM T53024 C3NYM8 42637137 IC50 > 1000 nM T53024 CJ47CL 42637210 IC50 > 1000 nM T53024 CR3A8Q 42637283 IC50 > 1000 nM T53024 CENZ47 42637363 IC50 > 1000 nM T53024 CX0JC7 42637503 IC50 > 1000 nM T53024 C90LHS 42637563 IC50 > 1000 nM T53024 C80WBK 42637632 IC50 > 1000 nM T53024 CR49YE 42637984 IC50 > 1000 nM T53024 CEFO24 42638065 IC50 > 1000 nM T53024 CF5JK4 42638066 IC50 > 1000 nM T53024 CJ06FD 44272606 Ki = 3.162 nM T53024 C71QSA 44272607 Ki = 1.259 nM T53024 CHY04A 44290718 IC50 = 1.3 nM T53024 C16BKW 44290734 IC50 = 3 nM T53024 CW76YB 44290735 IC50 = 4.1 nM T53024 CA6IS7 44290766 IC50 = 28.7 nM T53024 C6BZ1J 44298104 Ki = 81 nM T53024 CCXL10 44298113 Ki = 32 nM T53024 CYW8O0 44298130 Ki = 233 nM T53024 CB9JK1 44298131 Ki = 14 nM T53024 CJ5WL8 44298155 Ki = 99 nM T53024 CHL57J 44298156 Ki = 203 nM T53024 CP61LB 44298165 Ki = 16 nM T53024 CM0B6J 44298166 Ki = 37 nM T53024 C8XZR7 44298169 Ki = 69 nM T53024 C0DPX7 44298171 Ki = 163 nM T53024 C62OEU 44298177 Ki = 117 nM T53024 CS9JW8 44298178 Ki = 106 nM T53024 C20MBI 44298179 Ki = 31 nM T53024 C3QBP0 44298188 Ki = 633 nM T53024 C1R3QD 44298189 Ki = 32 nM T53024 C5RJ7U 44298195 Ki = 20 nM T53024 C8N3EJ 44298197 Ki = 51 nM T53024 CZU05A 44298214 Ki = 2230 nM T53024 CQUS98 44298218 Ki = 176 nM T53024 COTK07 44298219 Ki = 241 nM T53024 CAJO07 44298231 Ki = 543 nM T53024 C9S4IX 44298232 Ki = 76 nM T53024 CB1A3K 44298235 Ki > 1000 nM T53024 C2TQ1V 44298248 Ki = 637 nM T53024 C3WFV5 44298250 Ki = 16 nM T53024 CL2P9B 44298251 IC50 = 800 nM T53024 CVW19Y 44298328 Ki = 692 nM T53024 CT94HY 44298329 Ki > 1000 nM T53024 CL4F1V 44298378 Ki = 166 nM T53024 CMO1Q9 44298441 Ki = 12 nM T53024 C8Y9ZP 44298443 Ki = 25 nM T53024 CUSR45 44298468 Ki = 194 nM T53024 C8EN2H 44298469 Ki = 103 nM T53024 CWE7Q0 44298482 IC50 > 10000 nM T53024 CF69PL 44298522 Ki = 35 nM T53024 C3CHE2 44308782 Ki = 225 nM T53024 CBZH42 44308810 Ki = 1108 nM T53024 CU5S1P 44308833 Ki = 815 nM T53024 CRQJ98 44308836 Ki = 4 nM T53024 CRFM02 44308969 Ki = 1740 nM T53024 C40MJU 44308970 Ki = 0.04 nM T53024 C9KR7Q 44309052 Ki = 20 nM T53024 C4YG1S 44311590 IC50 > 10000 nM T53024 CY0OV9 44311591 IC50 = 213 nM T53024 C29GQB 44311601 IC50 = 42.5 nM T53024 CC8DS0 44311602 IC50 > 10000 nM T53024 C5KST2 44311690 IC50 > 1000 nM T53024 C6N4MH 44311691 IC50 > 10000 nM T53024 CIR4G6 44311695 IC50 > 10000 nM T53024 CTG6X5 44311696 IC50 > 1000 nM T53024 C7Y8SF 44311697 IC50 > 10000 nM T53024 CK52MY 44311702 IC50 > 1000 nM T53024 CX39CV 44311703 IC50 > 10000 nM T53024 C5RM2A 44311730 IC50 > 10000 nM T53024 CBG70T 44311731 IC50 > 1000 nM T53024 CQH20F 44311765 IC50 > 1000 nM T53024 CZG4K6 44311836 IC50 > 10000 nM T53024 CWNP79 44311837 IC50 > 1000 nM T53024 CWSF38 44311868 IC50 > 1000 nM T53024 C2T0YP 44311869 IC50 = 556 nM T53024 C1ONB3 44311870 IC50 = 343 nM T53024 C1GY0F 44311912 IC50 > 10000 nM T53024 C14DIH 44311913 IC50 > 10000 nM T53024 C1X4TI 44311914 IC50 = 43.8 nM T53024 C64WAE 44311958 IC50 > 1000 nM T53024 CFT90E 44311959 IC50 > 1000 nM T53024 C3PQD0 44311960 IC50 > 10000 nM T53024 CS7PB4 44312258 IC50 > 10000 nM T53024 C5PE1D 44325273 IC50 = 275 nM T53024 CQ1O9R 44325409 IC50 = 9.2 nM T53024 C2UO4D 44325410 IC50 = 6.9 nM T53024 CGS7C1 44325411 IC50 = 67 nM T53024 COW23D 44325425 IC50 = 3.2 nM T53024 CH0S5Q 44325451 IC50 = 85 nM T53024 C8CK2G 44325452 IC50 = 4.1 nM T53024 CZO9N5 44325456 IC50 > 2000 nM T53024 CL1HW3 44325477 IC50 = 6.5 nM T53024 CI17GX 44325478 IC50 = 2.9 nM T53024 C1P0QV 44332931 Ki > 10000 nM T53024 CM0SO4 44354260 Ki = 47 nM T53024 C41YZN 44354261 Ki = 10 nM T53024 CHJ6A4 44354297 Ki = 2.3 nM T53024 CL9A6X 44354298 Ki = 5.7 nM T53024 CAG1Z4 44354386 Ki = 120 nM T53024 C3QZH1 44354398 Ki = 15 nM T53024 C3KS5A 44354415 Ki = 2.5 nM T53024 CY5M4L 44354462 Ki = 8.6 nM T53024 C3NUG1 44354503 Ki = 95 nM T53024 C3R5VK 44354504 Ki = 5 nM T53024 C5YGJ4 44354505 Ki = 2.9 nM T53024 C5AGJ0 44354527 Ki = 17 nM T53024 CU20VL 44354528 Ki = 10 nM T53024 CYN83Q 44354529 Ki = 12 nM T53024 C6XB5J 44354552 Ki = 31 nM T53024 COB9V3 44354584 Ki = 21 nM T53024 C3NRE7 44354585 Ki = 5 nM T53024 C1IA4F 44354586 Ki = 2.8 nM T53024 C3MW4Q 44354587 Ki = 7.2 nM T53024 C51VDC 44354612 Ki = 9 nM T53024 CWZ08U 44354613 Ki = 11 nM T53024 C5QNB7 44354614 Ki = 35 nM T53024 CE3V2Z 44354615 Ki = 14 nM T53024 CR2T0L 44354649 Ki = 23 nM T53024 CC3W1P 44354650 Ki = 11 nM T53024 CI87FE 44354651 Ki = 178 nM T53024 C4QC6U 44354689 Ki = 23 nM T53024 CG7E3K 44354849 Ki = 85 nM T53024 C7KWL9 44354850 Ki = 4.6 nM T53024 CDN8O4 44354851 Ki = 85 nM T53024 C71AVO 44354852 Ki = 36 nM T53024 C1AU0K 44355050 Ki = 11 nM T53024 CVR20K 44355051 Ki = 10 nM T53024 CX1Y9V 44361984 Ki > 300000 nM T53024 C6UV4B 44362068 Ki = 4600 nM T53024 CHP41F 44363816 Ki = 3.6 nM T53024 CBPU86 44363919 Ki = 1.3 nM T53024 C19LVE 44363953 Ki = 80 nM T53024 CD9JY0 44363954 Ki = 6.3 nM T53024 C7N8RQ 44363956 Ki = 18 nM T53024 CN7E3K 44363998 Ki = 14 nM T53024 CWO13M 44363999 Ki = 47 nM T53024 CU1SK8 44364006 Ki = 122 nM T53024 CR7G6L 44364007 Ki = 40 nM T53024 CTC61E 44364008 Ki = 1.1 nM T53024 CHT0A8 44364016 Ki = 1.4 nM T53024 CI63XR 44364017 Ki = 12 nM T53024 CW7Y0A 44364027 Ki = 5.9 nM T53024 CLTH30 44364080 Ki = 2.2 nM T53024 C5T6VQ 44364081 Ki = 1 nM T53024 CPC5Q0 44364113 Ki = 4.6 nM T53024 CEC5V9 44364114 Ki = 11 nM T53024 CX6B7Z 44364115 Ki = 7.3 nM T53024 CH2DN4 44367916 IC50 > 10000 nM T53024 CM9YQ0 44367953 IC50 > 1000 nM T53024 C5W4YL 44368019 IC50 = 374 nM T53024 CO6ZJ9 44368020 IC50 = 474 nM T53024 CQ5T1D 44368043 IC50 = 204 nM T53024 C1SWO5 44368044 IC50 = 673 nM T53024 C29EZK 44368080 IC50 = 26 nM T53024 C9ZW6U 44368093 IC50 = 357 nM T53024 C71URM 44368094 IC50 = 16 nM T53024 CC1ZP9 44368109 IC50 > 1000 nM T53024 CQ7OP1 44368112 IC50 = 102 nM T53024 C0EW4I 44368117 IC50 = 22 nM T53024 C6TNZ9 44368144 IC50 > 1000 nM T53024 C53IAG 44368153 IC50 = 12 nM T53024 CKU8J7 44368156 IC50 = 130 nM T53024 CR12GB 44368157 IC50 = 41 nM T53024 C50DMO 44368226 IC50 = 575 nM T53024 CN31HS 44368398 IC50 = 594 nM T53024 C2RC0P 44368406 IC50 > 1000 nM T53024 CB1HC8 44368422 IC50 > 10000 nM T53024 C27DLY 44368489 IC50 > 1000 nM T53024 CWHK38 44377332 Ki > 10000 nM T53024 CVH1O7 44377366 Ki > 5000 nM T53024 CRC2N1 44377555 Ki = 2100 nM T53024 CS1WT5 44377591 Ki = 3200 nM T53024 C3LUY8 44377623 Ki > 10000 nM T53024 CQD0P4 44377645 Ki > 5000 nM T53024 CWNF42 44385504 Ki = 4220 nM T53024 CAFD79 44385508 Ki > 10000 nM T53024 CHY14B 44385591 Ki > 10000 nM T53024 CJQI19 44385652 Ki = 8680 nM T53024 CG12HD 44385712 Ki > 10000 nM T53024 C8MU5C 44385757 Ki = 5920 nM T53024 C0LRT9 44386389 Ki = 6040 nM T53024 C1EVK8 44387399 Ki = 345 nM T53024 C6U9VC 44388027 IC50 > 1000 nM T53024 C2IW5J 44388028 IC50 > 1000 nM T53024 C27ANT 44388029 IC50 > 1000 nM T53024 CHQK20 44388035 IC50 > 1000 nM T53024 CI9XS1 44388036 IC50 > 1000 nM T53024 CD4BX6 44388037 IC50 > 1000 nM T53024 CDS08Z 44388038 IC50 > 1000 nM T53024 CZA03Y 44388040 IC50 > 1000 nM T53024 C21WBR 44388043 IC50 > 1000 nM T53024 C7VK6B 44388052 IC50 > 1000 nM T53024 CT93BI 44388060 IC50 > 1000 nM T53024 C4E5VS 44388061 IC50 > 1000 nM T53024 C7P5RO 44388066 IC50 > 1000 nM T53024 C7T8IY 44388069 IC50 > 1000 nM T53024 C2TWO3 44388070 IC50 > 1000 nM T53024 CDBE87 44388075 IC50 > 1000 nM T53024 C25GWK 44388078 IC50 > 1000 nM T53024 CT93LV 44388079 IC50 > 1000 nM T53024 CX54SC 44388083 IC50 > 1000 nM T53024 C2C0RU 44388084 IC50 > 1000 nM T53024 C5SMA2 44388085 IC50 > 1000 nM T53024 C26OCG 44388086 IC50 > 1000 nM T53024 C8SR2O 44388087 IC50 > 1000 nM T53024 CHL5T1 44388088 IC50 > 1000 nM T53024 C4VNC2 44388089 IC50 > 1000 nM T53024 C1IH3T 44388090 IC50 > 1000 nM T53024 CNC91I 44388093 IC50 > 1000 nM T53024 CN45OF 44388095 IC50 > 1000 nM T53024 C82HJL 44388104 IC50 > 1000 nM T53024 CV6T2H 44388105 IC50 > 1000 nM T53024 CLC0N2 44388106 IC50 > 1000 nM T53024 C0VO1K 44388107 IC50 > 1000 nM T53024 CM5O3B 44388108 IC50 > 1000 nM T53024 CAF02P 44388109 IC50 > 1000 nM T53024 C23XBM 44388110 IC50 > 1000 nM T53024 CPX74G 44388112 IC50 > 1000 nM T53024 CG9SA3 44388114 IC50 > 1000 nM T53024 C2C4MH 44388116 IC50 > 1000 nM T53024 CW1EL5 44388118 IC50 > 1000 nM T53024 CN0K3V 44388119 IC50 > 1000 nM T53024 CE8DH4 44388120 IC50 > 1000 nM T53024 C1A0OY 44388121 IC50 > 1000 nM T53024 CS53NP 44388122 IC50 > 1000 nM T53024 CX67WG 44388123 IC50 > 1000 nM T53024 CB50EK 44388124 IC50 > 1000 nM T53024 C9SN1X 44388132 IC50 > 1000 nM T53024 C6W4YT 44388133 IC50 > 1000 nM T53024 CMTN20 44388134 IC50 > 1000 nM T53024 CAK42W 44388135 IC50 > 1000 nM T53024 CTW48B 44388136 IC50 > 1000 nM T53024 C4P1AS 44388137 IC50 > 1000 nM T53024 CEAZ82 44388138 IC50 > 1000 nM T53024 CZ2K1I 44397385 Ki = 32 nM T53024 C1KMT8 44397389 Ki = 2.7 nM T53024 C83JNK 44397472 Ki = 12 nM T53024 CE6U2K 44397620 Ki = 12 nM T53024 CM1W3L 44397628 Ki = 100 nM T53024 CN6Z8C 44397648 Ki = 4 nM T53024 CRW0M6 44397706 Ki = 1.8 nM T53024 CL7GX3 44397725 Ki = 610 nM T53024 C30MBR 44397747 Ki = 250 nM T53024 CQ0M7K 44397788 Ki = 220 nM T53024 C3MG9D 44397815 Ki = 2800 nM T53024 CK19EU 44397834 Ki = 640 nM T53024 C0OZB8 44397835 Ki = 5.6 nM T53024 C7X2VS 44397875 Ki = 430 nM T53024 C9DMA7 44397907 Ki = 160 nM T53024 CAD5S1 44397924 Ki = 23 nM T53024 C20TXF 44397990 Ki = 150 nM T53024 CM1R8X 44400000 IC50 = 11 nM T53024 CP89CS 44400135 IC50 = 0.2 nM T53024 CV4PO0 44403186 IC50 = 1.6 nM T53024 C8MEP3 44403194 IC50 = 6.2 nM T53024 C9B3AP 44403195 IC50 = 0.63 nM T53024 C29GND 44403204 IC50 = 11 nM T53024 CM3KG6 44403206 IC50 = 1.9 nM T53024 C0DG2C 44403217 IC50 = 1.4 nM T53024 C9MBD4 44403227 IC50 = 17 nM T53024 CLH53T 44403242 IC50 = 12 nM T53024 CIEM04 44403248 IC50 = 1.1 nM T53024 C1BY2P 44444935 IC50 = 44 nM T53024 CH17TI 44560858 IC50 = 3.6 nM T53024 C2AZY7 44560859 IC50 = 1.5 nM T53024 C2I8NB 44560860 IC50 = 0.75 nM T53024 C4XRT0 44560861 IC50 = 2.6 nM T53024 C21TZI 44560862 IC50 = 1.3 nM T53024 C2YM5N 44560863 IC50 = 2.7 nM T53024 CS39FB 44560864 IC50 = 5.7 nM T53024 CU3FD2 44560865 Ki = 5.51 nM T53024 C8IKU1 44560866 IC50 = 17 nM T53024 CTQ83Z 44560867 IC50 = 158 nM T53024 CQC29N 44560868 IC50 = 58 nM T53024 C47MDA 44560869 IC50 = 6.9 nM T53024 CHAJ41 44560870 IC50 = 23 nM T53024 CT0A9U 44560871 IC50 = 9.8 nM T53024 CM0T9R 44560872 IC50 = 46 nM T53024 CO2J6R 44560873 IC50 = 40 nM T53024 CKQD64 44560874 IC50 = 5.9 nM T53024 CEK26Y 44560875 IC50 = 4.1 nM T53024 CBL1P7 44560876 IC50 = 27 nM T53024 CY47DM 44560877 IC50 = 5.4 nM T53024 C5OZD1 44560878 IC50 = 15 nM T53024 CFT47C 44560898 IC50 = 52 nM T53024 CAO7R0 44560899 IC50 = 9.3 nM T53024 C80ZCF 44560900 IC50 = 9.3 nM T53024 CATH94 44560901 IC50 = 4.9 nM T53024 C2AXG6 44560902 IC50 = 23 nM T53024 COQ9W7 44560903 IC50 = 3.7 nM T53024 CLZ23V 44560904 IC50 = 1.4 nM T53024 C0OKG2 44560905 IC50 = 2.4 nM T53024 CPIW17 44560906 IC50 = 1.7 nM T53024 CFR3Y5 44560907 IC50 = 0.7 nM T53024 CS85LR 44560908 IC50 = 1.2 nM T53024 C6K1FI 44577218 IC50 = 337 nM T53024 CAJ15T 44577219 IC50 = 4.9 nM T53024 CQD56E 44577220 IC50 = 5.7 nM T53024 CV18IC 44577221 IC50 = 267 nM T53024 CLJD09 45102042 IC50 = 3320 nM T53024 C63YJS 45139239 IC50 = 44 nM T53024 C63XPN 45267999 IC50 > 1000 nM T53024 CF09UA 45268875 IC50 > 1000 nM T53024 C2PNH4 45272264 IC50 > 1000 nM T53024 CFL9K7 45273129 IC50 = 5.7 nM T53024 C9Z4MR 45273130 IC50 = 240 nM T53024 C4RGN0 45273131 IC50 = 100 nM T53024 CH18QA 46882131 Ki > 10000 nM T53024 CBZ3T9 46882132 Ki > 10000 nM T53024 C6KBJ2 46882133 Ki > 10000 nM T53024 CNL16U 46882180 Ki > 10000 nM T53024 CCX75M 46882181 Ki > 10000 nM T53024 C2BOJ6 46882182 Ki > 10000 nM T53024 C9ASC1 46882224 Ki > 10000 nM T53024 CB38SE 46882225 Ki > 10000 nM T53024 CP2N1U 46882226 Ki > 10000 nM T53024 CJ3Q6B 46882227 Ki > 10000 nM T53024 CRYQ47 46882445 Ki > 10000 nM T53024 CRZ1B0 46882446 Ki > 10000 nM T53024 CNEZ46 46882447 Ki > 10000 nM T53024 C8D1OR 46882448 Ki > 10000 nM T53024 CZ0G2R 46882449 Ki > 10000 nM T53024 CR37UF 46882513 Ki > 10000 nM T53024 CF3L8U 46882514 Ki > 10000 nM T53024 C91WKZ 46882515 Ki > 10000 nM T53024 CX21JH 46882516 Ki > 10000 nM T53024 CBJ92C 46882517 Ki > 10000 nM T53024 C8N3KX 46882577 Ki > 10000 nM T53024 CAH31I 46882578 Ki > 10000 nM T53024 CD2NL0 46882579 Ki > 10000 nM T53024 C9B0DF 46882620 Ki > 10000 nM T53024 CJ8I4L 46882621 Ki > 10000 nM T53024 C2YMA7 46882622 Ki > 10000 nM T53024 CD0VH7 46882664 Ki > 10000 nM T53024 C50YRJ 46882665 Ki > 10000 nM T53024 CXFV62 46882666 Ki > 10000 nM T53024 CR07WV 46882667 Ki > 10000 nM T53024 CF1HC7 46882668 Ki > 10000 nM T53024 CVIU56 46882708 Ki > 10000 nM T53024 C8S4LN 46882709 Ki > 10000 nM T53024 CJ7GM9 46882746 Ki > 10000 nM T53024 C6OM5H 46882789 Ki > 10000 nM T53024 C5MV8K 46882790 Ki > 10000 nM T53024 C6RD3V 46882791 Ki > 10000 nM T53024 C1WUF9 46882831 Ki > 10000 nM T53024 C5LM3W 46882832 Ki > 10000 nM T53024 CU1D6I 46902023 IC50 = 650 nM T53024 C84ZTC 49865341 IC50 = 44 nM T53024 C3VZ4U 49865342 IC50 > 1000 nM T53024 CGYR09 49865343 IC50 = 46 nM T53024 C35WID 49865344 IC50 = 9.6 nM T53024 C0RK7G 49865345 IC50 = 355.5 nM T53024 C4YLM7 49865346 IC50 = 87 nM T53024 CZ4RI1 49865347 IC50 = 101 nM T53024 CZ3E6D 52936625 Ki = 0.13 nM T53024 C2Z8US 52936721 Ki = 0.27 nM T53024 CJC1X5 52936722 Ki = 0.6 nM T53024 CVH8P1 52936723 Ki = 0.65 nM T53024 CXG57W 52936724 Ki = 0.13 nM T53024 C4RJ6K 52936725 Ki = 0.025 nM T53024 CJ63XR 52936830 Ki = 0.13 nM T53024 CK2S8L 52936831 Ki = 0.13 nM T53024 C92EDX 52936833 Ki = 0.025 nM T53024 C9SNL1 52941607 IC50 = 6100 nM T53024 C40ZRY 52948630 IC50 > 10000 nM T53024 C19ILO 53324674 IC50 = 0.4 nM T53024 C8Q7PC 53324675 IC50 > 600 nM T53024 CED3O6 53473658 IC50 = 35 nM T53024 CE7J0U 53473659 IC50 = 4.1 nM T53024 CY0G2K 53473744 IC50 = 15 nM T53024 CBQG96 53473824 IC50 = 1.6 nM T53024 CW53YV 53473917 IC50 > 1000 nM T53024 C87SME 53474004 IC50 = 106 nM T53024 C7EO1Z 53474005 IC50 > 1000 nM T53024 CY3M2A 53474090 IC50 > 1000 nM T53024 CEN8Y7 54580404 Ki = 1.5 nM T53024 CWM12T 54582417 Ki = 1400 nM T53024 CF3ED5 54584354 Ki = 20 nM T53024 CH76VW 54586271 Ki = 0.062 nM T53024 CPU92R 54586272 Ki = 0.18 nM T53024 CGKP76 56661222 Ki = 1 nM T53024 C3RWH0 56661224 Ki = 1 nM T53024 C9JHI4 56664813 Ki = 0.25 nM T53024 C3M6AT 56678313 Ki = 6.3 nM T53024 C05RSG 56681656 Ki > 1000 nM T53024 C59PKT 56681657 Ki > 0.07 nM T53024 C8ZW3O 56927659 IC50 = 4025 nM T53024 CHK8T1 56945132 Ki > 10000 nM T53024 C73XBL 57384077 IC50 > 1000 nM T53024 C3KC9Z 57398462 IC50 = 2.1 nM T53024 CH3IQ4 58723795 IC50 = 0.2 nM T53024 CHI36A 58723865 IC50 = 0.2 nM T53024 CTVI05 70683416 IC50 > 1000 nM T53024 CV42WQ 70689221 IC50 = 455 nM T53024 C3P0AN 70689413 IC50 = 5.5 nM T53024 CP58HL 70689414 IC50 = 4.4 nM T53024 CB14OW 70689415 IC50 = 3.1 nM T53024 CNZC97 70689723 IC50 > 1000 nM T53024 C2WQM9 70691295 IC50 > 1000 nM T53024 CIQ85K 70692642 Ki = 0.5 nM T53024 C5E8MY 70693613 IC50 = 4.1 nM T53024 C3TZ9U 70695246 IC50 = 509 nM T53024 C34XGS 70695722 IC50 = 45 nM T53024 CIPF50 70695723 IC50 = 4.2 nM T53024 CF08XL 71458043 Ki = 8600 nM T53024 CU82HG 71460000 IC50 > 10000 nM T53024 CPC69G 71461645 Ki = 6000 nM T53024 CLAV92 71461684 IC50 > 1000 nM T53024 C1NZU3 71461685 IC50 > 1000 nM T53024 C9J0EH 71603917 IC50 = 4100 nM T53024 CFKH42 71717904 IC50 = 37.6 nM T53024 CGDO59 72947672 Ki = 0.41 nM T53024 CW83DK 73213196 Ki > 10000 nM T53024 CIO28F 73345407 Ki = 17.1 nM T53024 CMN6X8 73345525 IC50 > 1000 nM T53024 C70XZC 73345528 IC50 = 24 nM T53024 CXGJ67 73345700 IC50 = 1.6 nM T53024 CV23JS 73345701 IC50 = 2 nM T53024 C81UME 73345740 Ki = 418 nM T53024 CX5VM1 73346900 IC50 > 1000 nM T53024 CA3MU5 73346903 IC50 = 0.33 nM T53024 CM08WH 73346925 Ki = 20 nM T53024 C62NFY 73346927 Ki = 810 nM T53024 CK64MX 73346930 Ki = 117 nM T53024 C15CAN 73346972 Ki = 6.98 nM T53024 CU2E9Z 73347200 EC50 = 1.7 nM T53024 CD09FU 73347225 Ki = 56 nM T53024 CI4L6W 73347226 Ki = 252 nM T53024 CGM61R 73348311 Ki > 10000 nM T53024 CN1FD2 73348312 Ki > 10000 nM T53024 C01GIQ 73348427 Ki = 89 nM T53024 C7Y9ZT 73348428 Ki = 317 nM T53024 CFLT50 73348719 IC50 = 8.4 nM T53024 C75NBQ 73348741 Ki = 35 nM T53024 C5MNX3 73348742 Ki = 84 nM T53024 CL94MY 73350006 Ki = 5.45 nM T53024 C0N6XK 73350010 Ki = 36 nM T53024 CTV30F 73350011 Ki = 51.8 nM T53024 CF2AK4 73350012 Ki = 24.7 nM T53024 CK9CS4 73351516 Ki = 9.33 nM T53024 CNY13O 73351517 Ki = 27.3 nM T53024 CUN6L1 73351622 IC50 = 173 nM T53024 CC98JE 73351624 IC50 = 57 nM T53024 CWUH52 73351718 Ki = 11.3 nM T53024 CS9I4W 73351829 Ki = 26 nM T53024 CF70XH 73351873 IC50 > 1000 nM T53024 C0KJ6N 73352984 Ki = 20 nM T53024 CFB54J 73352985 Ki = 12.1 nM T53024 CKFV85 73353009 Ki = 29.5 nM T53024 CC45AV 73353272 IC50 = 0.47 nM T53024 C41OCY 73353278 IC50 = 12.8 nM T53024 CW54CU 73353340 IC50 > 1000 nM T53024 CL7DT2 73354494 Ki = 1000 nM T53024 CA48EL 73354535 Ki = 2.33 nM T53024 CFK7Z3 73354633 IC50 = 339 nM T53024 C1UYL2 73354783 IC50 = 3.1 nM T53024 CG1CX0 73354798 IC50 = 2.5 nM T53024 CIVZ67 73354818 Ki = 12 nM T53024 CGCE64 73354819 Ki = 132 nM T53024 C1Y0CI 73356066 Ki = 197 nM T53024 C52JAS 73356068 Ki = 1000 nM T53024 CN5LG8 73356069 Ki = 189 nM T53024 C9GKV2 73356181 IC50 = 130 nM T53024 CG6RJ4 73356318 EC50 = 2.51 nM T53024 C7XFB6 73356331 IC50 = 5.2 nM T53024 CI02SE 73356366 Ki = 19 nM T53024 CW8L6C 76310862 IC50 = 946 nM T53024 CHV6K7 76314485 IC50 = 50 nM T53024 C0PR3Y 76314486 IC50 > 1000 nM T53024 C94BWD 76314487 IC50 = 1.6 nM T53024 C25XKO 76314488 IC50 = 0.76 nM T53024 CS54IV 76321777 IC50 = 11 nM T53024 C94OAT 76321778 IC50 = 1 nM T53024 CU1IR8 76325402 IC50 = 1.5 nM T53024 CL09JQ 86279005 IC50 > 10000 nM T53024 C3JOS4 86292350 Ki > 9600 nM T53024 CVLE34 86293506 Ki > 9590 nM T53024 C15VTO 86294248 Ki > 9600 nM T53024 C2BAV8 90644981 Ki = 311 nM T53024 CI58FM 90663867 IC50 = 2.2 nM T53024 CK62FO 90663868 IC50 = 1.2 nM T53024 C7AFD4 90663869 IC50 = 2 nM T53024 C4DM2Q 90663870 EC50 = 1.01 nM T53024 CS7U3P 90663871 EC50 = 2.13 nM T53024 C94XTF 90663872 IC50 = 1.1 nM T53024 CA7W0U 90663873 IC50 = 0.78 nM T53024 C4EG8T 90663874 IC50 = 0.95 nM T53024 CW21UO 90663875 IC50 = 2 nM T53024 CF71UB 90663876 EC50 = 1 nM T53024 C1EJ6Y 90663877 EC50 = 1.43 nM T53024 CA2LU6 90663878 EC50 = 1.12 nM T53024 C3T6QX 90663879 EC50 = 1.81 nM T53024 CRDV40 90663880 EC50 = 2.96 nM T53024 CI6L9F 90663881 EC50 = 2.62 nM T53024 C7Q4PD 90665458 Ki = 176000 nM T53024 CR43ZL 90665459 Ki = 198000 nM T53024 CLK7C3 90665460 Ki = 27000 nM T53024 CZ0UC6 90665461 Ki = 44000 nM T53024 C0IBJ6 90665462 Ki = 110000 nM T53024 CPX0C9 90665463 Ki = 55000 nM T53024 C3UVC8 91936728 IC50 = 2.5 nM T53024 CT3UP7 91936729 IC50 = 1.6 nM T53024 CD2E4L 101941290 IC50 = 7.8 nM T53024 C9KB3W 117711399 Ki > 9630 nM T53024 CTH52C 118718416 Ki = 0.5012 nM T53024 CKQ4P6 118718462 IC50 = 34.7 nM T53024 C1Z7UJ 118718463 Ki = 0.1995 nM T53024 CPYA80 118718465 IC50 = 2546 nM T53024 CR61UD 118718466 IC50 = 197 nM T53024 CW64XN 118718500 IC50 = 1812 nM T53024 CB4D5T 118718501 IC50 = 23.4 nM T53024 CW5HG2 118718502 IC50 = 355 nM T53024 CC36KP 118718503 IC50 = 17.8 nM T53024 C7FIQ1 118718504 IC50 = 824 nM T53024 CNBY57 118718505 IC50 = 669 nM T53024 CPY4Q5 118718506 IC50 = 35.3 nM T53024 CO13JR 118718507 IC50 = 435 nM T53024 CLFJ60 118718508 IC50 = 793 nM T53024 C13YUH 118718509 IC50 = 77.2 nM T53024 CP2O7U 118718510 IC50 = 526 nM T53024 CLDZ63 118718511 IC50 = 1000 nM T53024 CYQ7X2 118718854 IC50 = 533 nM T53024 CA6C4T 118719101 IC50 = 12 nM T53024 CDZ3H4 118719196 IC50 = 259 nM T53024 CQRO32 118719197 IC50 = 46 nM T53024 CGXH91 118719198 IC50 = 118 nM T53024 C1QJX7 118719199 IC50 = 29 nM T53024 C0GLC8 118719200 IC50 > 1000 nM T53024 C40NGQ 118719201 IC50 > 1000 nM T53024 CK2W9T 118719202 IC50 = 460 nM T53024 CW4AT0 118719275 IC50 > 1000 nM T53024 C5VWI1 118719303 IC50 = 82.9 nM T53024 CS12JW 122179457 IC50 > 10000 nM T53024 CNGQ19 122179477 IC50 > 100000 nM T53024 C6M3TH 127032865 Ki = 6850 nM T53024 CB5Q9D 127032866 Ki = 2660 nM T53024 CUO25F 127032867 Ki = 4690 nM T53024 CE79SV 138377584 IC50 > 10000 nM T53024 C9CEY3 145949026 Ki = 0.03 nM T53024 CG42NM 145964683 IC50 = 0.58 nM T53024 CAR6L2 145965091 IC50 = 2.6 nM T53024 C0UGS7 145965915 IC50 = 0.24 nM T53024 C6DIN9 145966680 IC50 = 0.6 nM T53024 CD73TX 145966884 IC50 = 0.68 nM T53024 C4YE5S 145973735 IC50 = 0.89 nM T53024 CSRI71 145974145 IC50 = 2 nM T53024 C5WM2G 145974146 IC50 = 0.69 nM T53024 CY0Z1U 145975165 IC50 = 0.31 nM T53024 C2X9MU 145975556 IC50 = 0.98 nM T53024 CCD0X3 145975716 IC50 = 2.3 nM T53024 CQX10C 145976310 IC50 = 2.3 nM T53024 CO6L5J 145977604 IC50 = 2.8 nM T53024 CNM36E 145977748 IC50 = 2.1 nM T53024 CYA13K 145977784 IC50 = 2 nM T53024 CZ98YX 145978229 IC50 = 1.8 nM T53024 C3E2GY 145978640 IC50 = 1.1 nM T53024 C0I2UD 155513010 Ki > 10000 nM T53024 CV2BZ9 155516168 Ki > 10000 nM T53024 C2OG9Y 155517592 Ki > 10000 nM T53024 C1BS2T 155519582 Ki > 10000 nM T53024 CHJO90 155524485 Ki > 10000 nM T53024 CI9HE4 155532172 Ki > 10000 nM T53024 CKZ82R 155538553 Ki > 10000 nM T53024 CBD2Q8 155541853 Ki = 0.68 nM T53024 COT04J 155544425 Ki = 0.022 nM T53024 CM0JT4 155546353 Ki = 0.12 nM T53024 C1E2QZ 155547005 Ki = 0.77 nM T53024 C08BZM 155548259 Ki = 0.19 nM T53024 CUVQ94 155550944 Ki = 0.12 nM T53024 C0C3FM 155551297 Ki = 0.015 nM T53024 CZ3IW6 155554285 Ki = 0.14 nM T53024 CN6S5M 155554925 Ki = 0.015 nM T53024 CX02AJ 155555535 Ki > 10000 nM T53024 CNA23E 155556911 Ki = 0.1 nM T53024 CR1AY2 155557409 Ki > 10000 nM T53024 CD58IO 155558366 Ki > 10000 nM T53024 C4FZC3 155559238 Ki = 0.14 nM T53024 CV5Q6F 155560117 Ki = 0.018 nM T53024 CP09EI 155561297 Ki = 0.075 nM T53024 C37MPB 155561497 Ki = 0.18 nM T53024 C96UIA 155562010 Ki = 0.015 nM T53024 C0OQY3 155563809 Ki = 0.97 nM T53024 C1PUW4 155565146 Ki = 0.26 nM T53024 CE27AD 155566365 Ki = 3350 nM T53024 CN7CQ1 155567326 Ki > 10000 nM T53024 COU5V6 155567788 Ki = 0.013 nM T53024 C9DW1Q 155569009 Ki = 0.061 nM T53024 CE76TG 42637005 IC50 > 1000 nM T53024 C6ELN4 42637006 IC50 > 1000 nM T53024 CS73LG 42637433 IC50 > 1000 nM T53024 C6C3YF 45270549 IC50 > 1000 nM T53024 C9Y3BS 45270550 IC50 > 1000 nM T53024 CQC51Z 45270552 IC50 > 1000 nM T53024 CXE30U 45271377 IC50 > 1000 nM T53024 D01BWV 9802572 Ki > 10000 nM T53024 D01NID 44388055 IC50 > 1000 nM T53024 D02CQW 11847438 IC50 = 3.6 nM T53024 D02IXC 44403231 IC50 = 18.6 nM T53024 D02NJV 44388048 IC50 > 1000 nM T53024 D02OJQ 44388115 IC50 = 16 nM T53024 D02WOX 44388129 IC50 > 1000 nM T53024 D03DRL 44388045 IC50 > 1000 nM T53024 D03SXC 44388041 IC50 > 1000 nM T53024 D03VHX 44388111 IC50 > 1000 nM T53024 D04EWA 44388034 IC50 > 1000 nM T53024 D04FPW 44388024 IC50 > 1000 nM T53024 D04ORV 44388047 IC50 = 15 nM T53024 D04QBM 5311374 Ki = 4720 nM T53024 D05COQ 11847588 IC50 = 2.2 nM T53024 D05XZA 44388071 IC50 > 1000 nM T53024 D06JWT 44388073 IC50 > 1000 nM T53024 D07DUF 44388130 IC50 > 1000 nM T53024 D07OSF 44388044 IC50 > 1000 nM T53024 D07WRP 15965425 Ki = 0.01 nM T53024 D09DAC 44388046 IC50 = 95 nM T53024 D09LHN 44311674 IC50 > 10000 nM T53024 D0A0DO 44388056 IC50 > 1000 nM T53024 D0A1XX 44388113 IC50 > 1000 nM T53024 D0BE3D 44388092 IC50 > 1000 nM T53024 D0C5RH 44388125 IC50 = 5 nM T53024 D0CC1P 44388042 IC50 > 1000 nM T53024 D0H0DC 44388051 IC50 > 1000 nM T53024 D0H4WH 44388128 IC50 = 43 nM T53024 D0I9ME 44388074 IC50 > 1000 nM T53024 D0J5OY 44388022 IC50 = 28 nM T53024 D0M5LA 44388050 IC50 = 598 nM T53024 D0N2MA 44388103 IC50 > 1000 nM T53024 D0N4LH 44388065 IC50 > 1000 nM T53024 D0O4GU 44403230 Ki = 1.7 nM T53024 D0P6ZZ 10581102 IC50 = 378 nM T53024 D0R0OX 44388102 IC50 > 1000 nM T53024 D0R4IS 44388131 IC50 > 1000 nM T53024 D0R7OD 44386062 Ki = 0.005 nM T53024 D0S7YR 44388059 IC50 > 1000 nM T53024 D0T5RO 16129706 Ki = 0.0016 nM T53024 D0W0AF 44388072 IC50 > 1000 nM T53024 D0WG0O 44388049 IC50 = 531 nM T53024 D0Z0OF 44388094 IC50 > 1000 nM T53024 D0Z1XY 44388064 IC50 > 1000 nM T53024 D0Z3LZ 44388023 IC50 = 1.9 nM T13714 D04LKS 25126798 Ki = 45000 nM T13714 D0G3PI 449171 EC50 = 1730 nM T13714 D0N0RU 82146 EC50 = 434 nM T13714 D00QWU 59251511 EC50 = 33 nM T13714 D0H4DR 49787490 EC50 = 0.6 nM T13714 D0L4FS 5280961 IC50 = 22000 nM T13714 D0R9YR 64971 EC50 > 50000 nM T13714 D0S5LT 29435 IC50 > 100000 nM T13714 D04XII 118883505 Ki = 160 nM T13714 D0TG1V 118883427 Ki = 1 nM T13714 D0W1XE 91827457 Ki = 1.3 nM T13714 CZ1D5B 4684 Ki = 169000 nM T13714 C8GBH5 7184 Ki = 66000 nM T13714 CUNQ92 7933 Ki = 184000 nM T13714 C3EA7W 13254 Ki = 62000 nM T13714 C6RWX2 16260 EC50 = 1008 nM T13714 CY7L2U 17570 Ki = 68000 nM T13714 C1BW7P 93017 EC50 > 50000 nM T13714 C5Q7RL 134528 EC50 = 85 nM T13714 C30ODV 246724 Ki = 476000 nM T13714 CE23KN 316046 EC50 = 1730 nM T13714 CT7A8Z 639844 Ki = 302000 nM T13714 C5T1DW 644851 EC50 = 640 nM T13714 C2EIZ4 680534 IC50 > 30000 nM T13714 CY6W1Z 912792 EC50 = 2573 nM T13714 CZ6Q1Y 1734080 IC50 = 175 nM T13714 C1YK9J 4585579 EC50 = 2637 nM T13714 CO76JI 4730488 EC50 = 245 nM T13714 CF58OK 5188108 EC50 = 180 nM T13714 C54OLI 5288679 EC50 = 40 nM T13714 C16ZSG 6439929 EC50 = 3600 nM T13714 C6R3GO 6539523 EC50 = 850 nM T13714 CX0A3D 7147072 Ki = 225000 nM T13714 C35IYW 8001903 EC50 = 530 nM T13714 C4QM3A 9808622 EC50 = 145 nM T13714 CD3CZ1 9817887 EC50 > 50000 nM T13714 CSP19Z 9930940 EC50 = 690 nM T13714 CI7CS1 10001458 IC50 = 100 nM T13714 CV7SK8 10064801 IC50 = 18000 nM T13714 C3HTA2 10070833 IC50 = 190 nM T13714 C2F4KU 10112384 IC50 = 20 nM T13714 C5NJP2 10129169 EC50 = 15 nM T13714 CG0LQ8 10129170 EC50 = 41 nM T13714 C18VCL 10196830 EC50 = 86 nM T13714 CSDA25 10218669 EC50 = 63 nM T13714 CF9PG8 10218693 EC50 = 25 nM T13714 C91PIS 10218694 EC50 = 87 nM T13714 CWOR09 10252443 IC50 = 180 nM T13714 C6Q0EM 10312252 EC50 = 145 nM T13714 C0GXN7 10312324 EC50 = 15 nM T13714 C4HDK8 10342621 IC50 = 130 nM T13714 CQ6R0U 10431545 IC50 = 170 nM T13714 CI34YL 10433666 IC50 = 20 nM T13714 CLP71Z 10528213 IC50 = 14000 nM T13714 C71EUS 11169139 IC50 = 7.8 nM T13714 C0Q8NA 11180636 EC50 = 26 nM T13714 CQGU73 11191949 IC50 = 2.4 nM T13714 C4DW7B 11261037 EC50 = 186 nM T13714 CK9V6O 11273187 EC50 = 12 nM T13714 C4JS1R 11352536 IC50 = 25 nM T13714 CS25IB 11360909 EC50 = 1400 nM T13714 C5XF7R 11377209 EC50 = 7 nM T13714 CPGA59 11489411 EC50 = 15 nM T13714 CRAZ96 11496708 EC50 = 20 nM T13714 C6CR9V 11503359 IC50 = 40 nM T13714 C0MX6B 11525365 EC50 = 650 nM T13714 C68RSH 11525752 EC50 = 700 nM T13714 CEDS09 11555148 EC50 = 160 nM T13714 CXV3T1 11555706 IC50 > 15000 nM T13714 CYS53Q 11559891 EC50 = 2300 nM T13714 CC68LI 11574384 IC50 = 30 nM T13714 C40UZA 11576047 EC50 = 470 nM T13714 C3ITH1 11582802 EC50 = 200 nM T13714 CP53LK 11583743 IC50 = 13 nM T13714 CU0D9H 11584508 IC50 = 3 nM T13714 C7FD2W 11592304 IC50 = 20 nM T13714 C3D7KA 11604995 IC50 = 2000 nM T13714 CK03GD 11611604 EC50 = 90 nM T13714 CX35ZF 11617908 EC50 = 200 nM T13714 C8EP5Z 11619338 IC50 = 630 nM T13714 CQN62W 11626766 EC50 = 580 nM T13714 C4ZR8D 11627859 IC50 = 2 nM T13714 C2WU8Q 11632271 EC50 = 300 nM T13714 C5Y1GK 11633117 EC50 = 160 nM T13714 C0T4UI 11639715 EC50 = 200 nM T13714 CTW7E6 11655554 IC50 = 410 nM T13714 CN26HX 11655575 EC50 = 4400 nM T13714 CX2H4T 11655676 IC50 = 3 nM T13714 C0N7VQ 11661439 EC50 = 200 nM T13714 CC0PO9 11662127 EC50 = 260 nM T13714 CQ2M8V 11669781 EC50 = 450 nM T13714 C9CQZ7 11683023 EC50 = 80 nM T13714 C47YFZ 11696530 EC50 = 500 nM T13714 CHW8N7 11697813 IC50 = 190 nM T13714 CTP37R 11697907 EC50 > 50000 nM T13714 CXB9Q8 11698867 IC50 = 5 nM T13714 C7P8FY 11704978 IC50 = 199 nM T13714 CGK13J 11705301 IC50 = 350 nM T13714 CG4IW2 11713433 IC50 = 4 nM T13714 C0MIV8 11713676 EC50 = 300 nM T13714 CFRG03 11721039 IC50 = 7 nM T13714 C3BJQ6 11853545 EC50 = 8600 nM T13714 CJXH73 11853546 IC50 = 63000 nM T13714 CWFP80 11853793 EC50 = 3650 nM T13714 CPI3X0 11853795 IC50 = 57000 nM T13714 C9VCA1 11854313 IC50 = 24000 nM T13714 CQ47XY 11854314 IC50 = 44000 nM T13714 CBNC08 11854315 IC50 = 10000 nM T13714 CR4W3T 11854316 IC50 = 14000 nM T13714 CM9Q3O 11854570 EC50 = 6540 nM T13714 C4I2NG 11854572 IC50 = 85000 nM T13714 C5QL6N 11854573 IC50 = 46000 nM T13714 CSN35D 11855081 IC50 = 10000 nM T13714 CS0IL9 11855082 EC50 = 2780 nM T13714 CCJ1N2 11855620 EC50 = 3630 nM T13714 CZ80OQ 11855623 IC50 = 62000 nM T13714 CMF9T0 11855894 IC50 = 19000 nM T13714 CXZW51 11856960 EC50 = 1160 nM T13714 CGYJ27 11857210 IC50 = 12000 nM T13714 C7HN1R 11857214 IC50 = 42000 nM T13714 CKS09G 12949989 EC50 = 6152 nM T13714 C2V9RQ 13028610 EC50 = 1985 nM T13714 C7SC2A 13659563 Ki = 153000 nM T13714 CG7U2N 14239481 EC50 > 50000 nM T13714 C3HA7T 15953841 IC50 = 740 nM T13714 C43ZTW 16049406 IC50 = 170 nM T13714 CA1U0H 16049407 IC50 = 30 nM T13714 CFMX18 16049474 IC50 = 30 nM T13714 C8ZY3L 16049475 IC50 = 25 nM T13714 CK75FX 16049476 IC50 = 40 nM T13714 CCF48P 16049477 IC50 = 120 nM T13714 C46MDG 16049478 IC50 = 290 nM T13714 CC95QW 16049479 IC50 = 50 nM T13714 CPIM37 16049537 IC50 = 165 nM T13714 CH42EK 16049538 IC50 = 115 nM T13714 CU9G5E 16049539 IC50 = 45 nM T13714 C9D5TB 16049540 IC50 = 30 nM T13714 CEX8N2 16049541 IC50 = 30 nM T13714 C0DVS7 16072077 EC50 < 31622.78 nM T13714 CT32VG 16090326 EC50 = 296 nM T13714 CCT84J 16090327 EC50 = 1500 nM T13714 C03ZSF 16090328 EC50 = 1500 nM T13714 C28VIS 16090329 IC50 = 5 nM T13714 CF4J1K 16090330 IC50 = 1.9 nM T13714 CUR0Y7 16090331 IC50 = 7 nM T13714 C1IF8A 16090332 IC50 = 115 nM T13714 CL45DA 16718799 EC50 = 406 nM T13714 CKH5O1 16725052 EC50 = 12 nM T13714 C6NOS9 16727104 EC50 = 31 nM T13714 CXVS20 16727105 IC50 = 2.1 nM T13714 CN6CU3 16739344 IC50 = 5 nM T13714 CBUG37 17753624 EC50 = 60 nM T13714 C2LMW1 18565134 EC50 = 3800 nM T13714 C0QKH8 18565138 EC50 = 3200 nM T13714 CGS1R9 18565141 EC50 = 2600 nM T13714 CP3AS5 19835803 EC50 = 232 nM T13714 C38JEL 20704150 EC50 = 10 nM T13714 CWU4M0 20704168 IC50 > 10000 nM T13714 C6FGV5 20704187 IC50 = 2200 nM T13714 CZ0PC4 21037789 IC50 = 3800 nM T13714 CTE9J2 21050637 IC50 > 10000 nM T13714 C0FQ7Y 21943462 IC50 = 1500 nM T13714 C9MFJ3 21943465 IC50 = 700 nM T13714 C5M2BR 22042560 IC50 = 1700 nM T13714 CKQ7J8 22042567 IC50 = 1800 nM T13714 C5P2XM 22042570 IC50 = 600 nM T13714 C0FM4D 22042579 IC50 = 600 nM T13714 C26CJW 22042583 IC50 = 2500 nM T13714 CO6Y1G 22042586 IC50 = 8000 nM T13714 CL56EK 22042589 IC50 = 800 nM T13714 CZVR95 22042593 IC50 = 600 nM T13714 C1R9XS 22042597 IC50 = 8000 nM T13714 C9J0FI 22042604 IC50 = 4100 nM T13714 CY4TN3 22042608 IC50 = 1400 nM T13714 CC76YM 22042611 IC50 = 400 nM T13714 C19AML 22042616 IC50 = 300 nM T13714 C9O2XF 22042617 IC50 = 600 nM T13714 CGC2J5 22042622 IC50 > 10000 nM T13714 CWR7N6 22042624 IC50 = 1100 nM T13714 CPA92E 22042635 IC50 = 900 nM T13714 CIDN03 22042636 IC50 = 700 nM T13714 C25QOP 22042637 IC50 > 30000 nM T13714 CPJ6V3 22042638 IC50 = 1100 nM T13714 C0T1YA 22042641 IC50 = 600 nM T13714 C8AMJ5 22042645 IC50 = 500 nM T13714 C0IB6G 22042647 IC50 = 10000 nM T13714 CR0D8Q 22042652 IC50 = 600 nM T13714 C3BD4J 22042654 IC50 = 7500 nM T13714 C63JBD 22061016 Ki = 28000 nM T13714 CWD19A 23643871 EC50 = 98 nM T13714 C5W1QM 23648467 EC50 = 100 nM T13714 CL84DN 23648468 IC50 = 3.7 nM T13714 CZU9G4 23648469 IC50 = 56.4 nM T13714 C4J1KP 23648470 IC50 = 33.8 nM T13714 CF9E7D 23648471 IC50 > 10000 nM T13714 CT50PV 23648472 IC50 = 5.5 nM T13714 CUTE13 23648473 IC50 = 17 nM T13714 CR1JB8 23648474 IC50 = 154 nM T13714 CX6FT2 23648475 EC50 = 39 nM T13714 CS26KY 23648476 IC50 = 1.4 nM T13714 CRS43H 23648477 EC50 = 141 nM T13714 C6CAG2 23648478 IC50 = 12 nM T13714 CFG0L7 23648479 IC50 > 10000 nM T13714 CYA97J 23648480 IC50 = 138 nM T13714 C26XFS 23648481 EC50 = 58 nM T13714 CH6O5G 23648482 EC50 = 78 nM T13714 CY4I6V 23648483 EC50 = 4003 nM T13714 C2RJ1K 23648484 EC50 = 316 nM T13714 CO8M2W 23648485 IC50 = 5.4 nM T13714 CE1G7K 23648486 EC50 = 770 nM T13714 C03PJK 23648487 EC50 = 2304 nM T13714 CD1N3S 23648488 IC50 = 276 nM T13714 C0RCT4 23648532 EC50 = 63 nM T13714 CG2V6T 23648533 EC50 = 76 nM T13714 C30RES 23648534 EC50 = 200 nM T13714 CXOG70 23648535 EC50 = 35 nM T13714 CYL8W7 23648536 EC50 = 6 nM T13714 C9A4RZ 23648537 EC50 = 150 nM T13714 CJD4H1 23648538 EC50 = 800 nM T13714 CX5FC4 23648540 EC50 = 980 nM T13714 C6OM0B 23648541 EC50 = 560 nM T13714 CA25OJ 23648542 EC50 = 470 nM T13714 CIDA95 23648543 EC50 = 140 nM T13714 C1J5LG 23648544 EC50 = 170 nM T13714 CG8J3O 23648545 EC50 = 160 nM T13714 CU7BE2 23648546 EC50 = 81 nM T13714 CP91XL 23648547 EC50 > 10000 nM T13714 CA8CW9 23648548 EC50 = 3700 nM T13714 C6WX4P 23648549 EC50 = 3400 nM T13714 CY09RV 23648550 EC50 = 4000 nM T13714 CW0T7E 23648551 EC50 = 7700 nM T13714 C9XC1H 23648552 EC50 = 970 nM T13714 CG86DV 23648553 EC50 = 600 nM T13714 C01JZF 23648554 EC50 = 250 nM T13714 CTE1N2 24748569 EC50 > 10000 nM T13714 C06CYE 24764397 EC50 = 351 nM T13714 CW4Y9N 24767795 IC50 = 2000 nM T13714 CPJB16 24768116 EC50 = 70 nM T13714 CH58ID 24768117 EC50 = 110 nM T13714 C1ZJT0 24768118 EC50 = 200 nM T13714 CKJ8O1 24768119 EC50 = 260 nM T13714 CR7VX5 24768120 EC50 = 300 nM T13714 C7WA9T 24768121 EC50 = 560 nM T13714 CA52ER 24768122 EC50 = 575 nM T13714 C8N1RD 24776331 EC50 < 31622.78 nM T13714 C1U5CP 24776332 EC50 = 1584.89 nM T13714 C4W1LF 24776334 EC50 = 2511.89 nM T13714 C38CHU 24776335 EC50 < 31622.78 nM T13714 CTXB68 24776336 EC50 < 31622.78 nM T13714 C0TYF8 24776337 EC50 < 31622.78 nM T13714 CS0YZ8 24776338 EC50 = 3162.28 nM T13714 C0Z2OY 24776339 EC50 < 31622.78 nM T13714 C59ZYO 24776340 EC50 = 630.96 nM T13714 CP0GA4 24808559 EC50 = 500 nM T13714 C76BPI 24860506 IC50 = 12000 nM T13714 C5PJ0G 24860507 IC50 = 26000 nM T13714 C8C4ME 24860508 IC50 = 46000 nM T13714 C62QOY 24860509 IC50 = 41000 nM T13714 C67AFM 24860510 IC50 = 11000 nM T13714 CV1Q0H 24936142 IC50 = 5 nM T13714 C6ZG0A 24936147 EC50 = 4167 nM T13714 CC13ZW 24936148 IC50 = 15 nM T13714 C18VZL 24986297 EC50 = 1800 nM T13714 CL10IN 24986299 EC50 = 1100 nM T13714 CUV4C0 24986301 EC50 = 2800 nM T13714 CEA64D 24991075 EC50 = 1900 nM T13714 CO08HG 24991077 EC50 = 2000 nM T13714 CFJ34K 24991433 EC50 = 2200 nM T13714 C14HGJ 24991436 EC50 = 1800 nM T13714 CC0QH2 24991785 EC50 = 1800 nM T13714 CF1HS7 24991787 EC50 = 1900 nM T13714 CA1MU6 24991788 EC50 = 2700 nM T13714 CN6J4S 25099837 IC50 > 1000 nM T13714 CZW14K 25099838 IC50 = 61 nM T13714 CD9W8I 25099839 IC50 = 118 nM T13714 CN97XU 25099842 IC50 = 2.2 nM T13714 CCA5I2 25099990 IC50 = 4.7 nM T13714 CFPR78 25099991 IC50 = 19 nM T13714 CE5M6T 25100147 IC50 = 153 nM T13714 CS3ZP8 25100148 IC50 = 121 nM T13714 C83EZA 25100149 IC50 = 3.3 nM T13714 CY0V6M 25100150 IC50 = 1 nM T13714 CS87WP 25100151 IC50 = 6.6 nM T13714 CLA0E4 25100152 IC50 = 3.4 nM T13714 CR7EZ5 25100307 IC50 = 28 nM T13714 C4VF6J 25100311 IC50 = 2 nM T13714 CBOL78 25100472 IC50 = 40 nM T13714 CQSF65 25100922 IC50 = 4 nM T13714 CQL7E3 25102117 IC50 = 6.1 nM T13714 CPG4W6 25102118 IC50 = 23 nM T13714 C4ANQ0 25102119 IC50 = 7.9 nM T13714 CI4O1G 25102122 IC50 = 56 nM T13714 C0QD2M 25102124 IC50 = 1076 nM T13714 C7XW8B 25102125 IC50 = 2 nM T13714 CBY8K4 25107513 IC50 = 40 nM T13714 C3KC6G 25137978 EC50 = 990 nM T13714 CO80QT 25137979 EC50 = 2890 nM T13714 C08ANI 25137980 EC50 = 5720 nM T13714 C4WMH5 25137981 EC50 = 9050 nM T13714 CG87IF 25137982 EC50 = 9800 nM T13714 CU6YO2 25137983 IC50 = 30 nM T13714 CS3V8P 25137984 EC50 = 10200 nM T13714 C0DX5J 25137985 IC50 = 38 nM T13714 C87YAR 25137986 IC50 = 48 nM T13714 CB3CS4 25137987 IC50 = 1853 nM T13714 CB6J0R 25147499 EC50 = 4 nM T13714 CI2XO4 25190753 EC50 = 60 nM T13714 C5TQ2G 25190754 EC50 = 510 nM T13714 CN67OC 25190755 EC50 = 288 nM T13714 C5B4MW 25190756 EC50 = 23 nM T13714 CWS3O8 25190757 EC50 = 15 nM T13714 CF9C1A 25190793 EC50 = 420 nM T13714 C04QZS 25190794 EC50 = 120 nM T13714 CJG96H 25190795 EC50 = 220 nM T13714 COX5R7 25190796 EC50 = 350 nM T13714 CG9P2U 25190797 EC50 = 1320 nM T13714 CE1F0M 25190798 EC50 = 58 nM T13714 CCV8H1 25190800 EC50 = 1800 nM T13714 C0WK4E 25190801 EC50 = 1750 nM T13714 C01GPA 25190802 EC50 = 360 nM T13714 CLV9B7 25190803 EC50 = 5600 nM T13714 CEK8Y7 25190804 EC50 = 300 nM T13714 C4QBE2 25190806 EC50 = 380 nM T13714 CK5DU7 25190807 EC50 = 420 nM T13714 CHMP24 25190809 EC50 = 57 nM T13714 C53CGY 25190810 EC50 = 4900 nM T13714 C0ICK2 25190811 EC50 = 490 nM T13714 C5BU4J 25190812 EC50 = 1510 nM T13714 CD1SK4 25190813 EC50 = 1780 nM T13714 CB1M8E 25190814 EC50 = 1780 nM T13714 C5UQF2 25190815 EC50 > 30000 nM T13714 C8MY4C 25190816 EC50 > 30000 nM T13714 C6W8AT 25190817 EC50 > 30000 nM T13714 CYH9X7 25190818 EC50 > 30000 nM T13714 CEB2L5 25190819 EC50 = 1500 nM T13714 CON0T8 25190820 EC50 = 26000 nM T13714 C03ESA 25190821 EC50 = 28000 nM T13714 C75KAZ 25190822 EC50 = 18000 nM T13714 CZ3U1C 25190823 EC50 > 30000 nM T13714 C3P2QZ 25190824 EC50 = 1600 nM T13714 CB7GM1 25190825 EC50 = 300 nM T13714 C8FP4X 25190826 EC50 = 670 nM T13714 CNW2S9 25190827 EC50 = 660 nM T13714 C23PFA 25190828 EC50 = 130 nM T13714 CHS64Q 25190829 EC50 > 30000 nM T13714 C0CMB7 25190830 EC50 > 30000 nM T13714 CY31NZ 25190831 EC50 = 1600 nM T13714 CR27GM 25190832 EC50 = 1300 nM T13714 CNO3X8 25190833 EC50 = 1400 nM T13714 C2M3XZ 25190834 EC50 > 30000 nM T13714 C1PKR2 25190835 EC50 > 30000 nM T13714 C4GE9S 25190836 EC50 = 1160 nM T13714 CE8X5A 25190837 EC50 = 900 nM T13714 CZJ87X 25190838 EC50 = 2100 nM T13714 CX63NO 25190839 EC50 > 30000 nM T13714 CTG81N 25190840 EC50 > 30000 nM T13714 CN2MP4 25190841 EC50 > 30000 nM T13714 C1TQ4S 25190842 EC50 > 30000 nM T13714 CVX09K 25190843 EC50 > 30000 nM T13714 CU8GT2 25190844 EC50 > 30000 nM T13714 CVPH15 25190845 EC50 > 10000 nM T13714 CZ04FK 25190846 EC50 = 1160 nM T13714 CW4DI9 25190847 EC50 = 120 nM T13714 C5OMU2 25190848 EC50 = 650 nM T13714 CXHU40 25190849 EC50 = 430 nM T13714 CMTH65 25190850 EC50 = 730 nM T13714 CCAU42 25190851 EC50 = 1810 nM T13714 CYI08G 25190852 EC50 = 1330 nM T13714 CHRS63 25190853 EC50 = 960 nM T13714 CCT48R 25190854 EC50 = 460 nM T13714 CC5EV2 25190855 EC50 = 600 nM T13714 CN0O8M 25190856 EC50 = 3350 nM T13714 C2XD8T 25190857 EC50 = 200 nM T13714 C5WP3Y 25190858 EC50 = 600 nM T13714 CKNI08 25190859 EC50 = 800 nM T13714 CN4T9L 25190860 EC50 = 100 nM T13714 CX9TD7 25190861 EC50 = 52 nM T13714 CG35DI 25190862 EC50 = 760 nM T13714 CEDZ28 25190863 EC50 = 110 nM T13714 CHS74M 25190864 EC50 = 336 nM T13714 CGFY70 25190865 EC50 = 130 nM T13714 CVY5A6 25190866 EC50 = 2100 nM T13714 CQ3J0R 25190867 EC50 = 520 nM T13714 CKN73R 25190868 EC50 = 210 nM T13714 CG6A4T 25190869 EC50 = 400 nM T13714 CC8NZ3 25190870 EC50 = 190 nM T13714 CNI6S2 25190871 EC50 = 170 nM T13714 CYP1F3 25190872 EC50 = 470 nM T13714 C9JFS4 25190873 EC50 = 530 nM T13714 COI2X7 25190874 EC50 = 1500 nM T13714 C8DI4A 25210583 EC50 = 1 nM T13714 C14HCZ 25218828 EC50 = 250 nM T13714 CM4WA9 25218829 EC50 = 370 nM T13714 C5U2ED 25218830 IC50 = 31200 nM T13714 C2VFE6 25218831 IC50 = 150 nM T13714 CA0H5N 25218832 EC50 = 1530 nM T13714 CE7HR1 25218833 EC50 = 3160 nM T13714 CGY57P 25218834 EC50 = 1810 nM T13714 CUP27J 25218835 EC50 = 430 nM T13714 C1D7CS 25218836 IC50 = 56 nM T13714 CZ09XS 25218837 EC50 = 190 nM T13714 CWHJ63 25218838 EC50 = 360 nM T13714 CBV2X7 25218839 EC50 = 150 nM T13714 CPY79U 25218840 EC50 = 340 nM T13714 CKX1O5 25218841 EC50 = 270 nM T13714 CRA4T3 25218842 EC50 = 370 nM T13714 CF5BR4 25218843 EC50 = 400 nM T13714 CXN2U4 25218844 EC50 = 110 nM T13714 C4MWC5 25218845 EC50 = 170 nM T13714 C8W0TY 25218846 IC50 = 65 nM T13714 C7MU6E 25218847 EC50 = 92 nM T13714 CO95WI 25218848 EC50 = 76 nM T13714 CUS41I 25218849 EC50 = 210 nM T13714 CVF58N 25218851 EC50 = 120 nM T13714 C3UI9O 25225010 IC50 = 35 nM T13714 CWO5V0 25225786 IC50 = 3 nM T13714 CZ9CE5 25226691 IC50 = 4 nM T13714 CX3ID9 25226692 IC50 = 11 nM T13714 C9TJ4D 25226881 IC50 = 2 nM T13714 CQIB51 25227069 IC50 = 2 nM T13714 C4Q5BN 25227247 IC50 = 4 nM T13714 CS1EJ7 25234324 IC50 = 450 nM T13714 C0J4GU 25918963 Ki > 500000 nM T13714 CK9X5Z 37818370 Ki = 10000 nM T13714 C0VHF6 42601437 EC50 = 2600 nM T13714 CR09VW 42641405 EC50 = 144 nM T13714 C5BT2G 42641974 IC50 = 3.2 nM T13714 C53TKQ 44123769 EC50 = 138 nM T13714 C0J5LA 44135945 IC50 > 1000 nM T13714 CC41IF 44136012 IC50 = 44 nM T13714 CYEQ65 44136014 IC50 = 85 nM T13714 CD5N0Y 44136075 EC50 = 930 nM T13714 CWNG36 44136213 IC50 = 239 nM T13714 CP51NL 44136346 EC50 = 6500 nM T13714 C4E8PW 44136349 IC50 > 1000 nM T13714 C2V6PL 44136351 IC50 > 1000 nM T13714 C9Z3FW 44136417 IC50 = 34 nM T13714 CK0WE9 44136418 IC50 = 35 nM T13714 C7QRB9 44136419 IC50 = 45 nM T13714 CFI79Y 44136477 EC50 = 1660 nM T13714 C4OGJ0 44136604 EC50 = 3900 nM T13714 CJM3P2 44136717 EC50 = 2180 nM T13714 C9XS4G 44136902 IC50 = 128 nM T13714 C3SK9J 44136969 EC50 = 1110 nM T13714 CA87MH 44137029 IC50 = 248 nM T13714 C41PXG 44137030 IC50 = 489 nM T13714 CAN35S 44137031 IC50 = 315 nM T13714 CD0ET3 44137032 IC50 = 436 nM T13714 CP13OK 44137033 IC50 = 462 nM T13714 CIJA24 44137094 IC50 > 1000 nM T13714 C9IXQ3 44137098 IC50 > 1000 nM T13714 C8B9ZN 44137168 IC50 = 26 nM T13714 C90LGQ 44137229 IC50 > 1000 nM T13714 C0FDZ1 44137303 IC50 = 882 nM T13714 C9QR5C 44137304 IC50 = 22 nM T13714 CLTG76 44137366 IC50 = 799 nM T13714 CH8UB0 44137367 IC50 = 561 nM T13714 C9R0KB 44137369 IC50 > 1000 nM T13714 CNB45D 44137441 IC50 = 16 nM T13714 C5EL2Q 44137442 IC50 = 4.7 nM T13714 CW41UJ 44137443 IC50 = 93 nM T13714 CC9Y5H 44137444 IC50 = 2.6 nM T13714 C86AME 44137503 IC50 > 1000 nM T13714 C89GVM 44137575 IC50 = 5.1 nM T13714 C1GH4M 44137576 EC50 = 640 nM T13714 CH50TJ 44137636 EC50 = 1220 nM T13714 CW7IY5 44137712 IC50 = 6400 nM T13714 C5NFR2 44137713 IC50 = 100 nM T13714 C6R1UH 44137714 IC50 = 99 nM T13714 CHA73X 44137715 IC50 = 138 nM T13714 CF8D0P 44137845 IC50 = 183 nM T13714 CSO53M 44137979 IC50 = 14 nM T13714 C28EXH 44137980 IC50 = 12 nM T13714 CNVL89 44137982 IC50 = 36 nM T13714 CK8R4C 44180521 EC50 = 525 nM T13714 C37NLY 44217616 EC50 = 1400 nM T13714 CY8RX6 44217767 EC50 = 1100 nM T13714 CP0W5I 44218087 EC50 = 1200 nM T13714 COEB58 44399795 EC50 = 1 nM T13714 CHT2S3 44400184 IC50 = 29 nM T13714 C1XZ3Q 44400273 IC50 = 163 nM T13714 C2F7JU 44400646 EC50 = 2 nM T13714 C4FA9O 44400680 IC50 = 12 nM T13714 C3G2HU 44400748 EC50 = 1 nM T13714 CRWF17 44403557 IC50 = 420 nM T13714 CWT40V 44403558 EC50 = 70 nM T13714 CZT94C 44403564 EC50 = 1500 nM T13714 C5XQW3 44403565 EC50 = 100 nM T13714 CD9S3C 44403570 IC50 = 290 nM T13714 C8K9ZM 44403571 IC50 = 120 nM T13714 C9C2JX 44403589 IC50 = 1010 nM T13714 CTN5Z2 44403617 IC50 = 2900 nM T13714 C34OXW 44403619 IC50 > 15000 nM T13714 C31FVO 44403620 IC50 = 3850 nM T13714 CU4H2G 44403625 IC50 = 5000 nM T13714 C5V6GE 44403626 IC50 = 2220 nM T13714 CA2CW3 44403633 IC50 = 4120 nM T13714 CC7J1B 44403639 IC50 = 310 nM T13714 C38VRQ 44403645 IC50 = 200 nM T13714 COW1B4 44403655 IC50 = 530 nM T13714 CXPJ14 44403656 IC50 = 190 nM T13714 CZK0P5 44409123 IC50 > 10000 nM T13714 CW9S1K 44411622 IC50 = 428 nM T13714 CNL81R 44411653 IC50 = 65 nM T13714 CW3AV8 44411661 IC50 = 100 nM T13714 C4MAN2 44411789 IC50 = 140 nM T13714 CYJ25W 44411810 IC50 = 970 nM T13714 C8FBH9 44411838 IC50 = 170 nM T13714 C4U2SJ 44411842 IC50 = 25 nM T13714 CJF9L1 44411843 IC50 = 89 nM T13714 CX6DN0 44411977 EC50 = 3500 nM T13714 CP46GF 44412005 EC50 = 124 nM T13714 CBVJ21 44412006 EC50 = 1300 nM T13714 C8DPK5 44412188 IC50 = 320 nM T13714 CPK6G2 44412195 IC50 = 26 nM T13714 CEU76F 44416756 IC50 = 20 nM T13714 CR97GI 44416799 IC50 = 900 nM T13714 C3YB5A 44416802 EC50 = 400 nM T13714 CNC6B7 44416803 EC50 = 100 nM T13714 CK82QS 44416818 EC50 = 5400 nM T13714 CZN20F 44416819 EC50 = 11000 nM T13714 C0R2KB 44416821 EC50 = 100 nM T13714 C1SQM3 44416822 EC50 = 600 nM T13714 CL9HK1 44416842 IC50 = 500 nM T13714 CIXR07 44416843 IC50 = 32000 nM T13714 C6DU1G 44416861 IC50 = 90000 nM T13714 C2GD1Q 44416897 EC50 = 70 nM T13714 CZ1N4K 44416914 IC50 = 60 nM T13714 C4L7VQ 44416915 EC50 = 40 nM T13714 C53BAF 44416930 IC50 = 30 nM T13714 CW3NF9 44416950 EC50 = 700 nM T13714 CQHE10 44416951 EC50 = 200 nM T13714 CP8Y5T 44416988 EC50 = 2300 nM T13714 C5RB8X 44416991 IC50 = 31000 nM T13714 CDG8Z0 44416992 EC50 = 2400 nM T13714 C6MEG2 44417023 IC50 = 1200 nM T13714 CPSL50 44417026 EC50 = 260 nM T13714 CR82JZ 44417027 IC50 = 20 nM T13714 CWDI21 44417028 EC50 = 1200 nM T13714 CB6LY0 44417045 EC50 = 2300 nM T13714 CKR1H6 44417046 EC50 = 30 nM T13714 COX48N 44417052 EC50 = 300 nM T13714 C1TH7E 44417068 IC50 = 40 nM T13714 CAJH47 44417072 IC50 = 50 nM T13714 CL50IQ 44423673 EC50 = 286 nM T13714 CAS1M0 44428685 EC50 = 3981.07 nM T13714 C5YT0R 44432612 EC50 = 230 nM T13714 CQK4F0 44446235 IC50 = 5 nM T13714 C6E8BG 44446237 IC50 = 67 nM T13714 CGI9W5 44446239 IC50 = 81 nM T13714 CC29YZ 44446242 IC50 = 473 nM T13714 C34HCM 44446244 IC50 = 5 nM T13714 CAK9X2 44446246 IC50 = 2 nM T13714 C65ZXY 44446249 IC50 = 10 nM T13714 CZ2T6A 44446253 IC50 = 219 nM T13714 C6GR7Q 44446254 IC50 = 26 nM T13714 CEDU42 44472980 EC50 = 895 nM T13714 C5OUG9 44472981 EC50 = 1030 nM T13714 CTZ48C 44472982 IC50 = 14 nM T13714 C0FJT4 44472983 EC50 = 646 nM T13714 CK3H2I 44472984 EC50 = 1010 nM T13714 CO8FG1 44472985 EC50 = 3400 nM T13714 CR0Q7O 44472986 IC50 > 1000 nM T13714 CX18UB 44472987 EC50 = 1370 nM T13714 CN30ED 44472988 IC50 = 230 nM T13714 C41NFW 44472989 IC50 = 12 nM T13714 CI92RZ 44472990 EC50 = 108 nM T13714 CO7U1F 44472991 EC50 = 612 nM T13714 CS8EI5 44472992 EC50 = 1525 nM T13714 CC3KU9 44472993 IC50 = 10 nM T13714 CZO32E 44472994 EC50 = 144 nM T13714 CTI06D 44472995 EC50 = 98 nM T13714 C69VFJ 44472996 IC50 = 2.9 nM T13714 CE58LO 44472997 IC50 = 125 nM T13714 C6U0PL 44472998 EC50 = 1272 nM T13714 CKB13G 44472999 EC50 = 1180 nM T13714 CKOR84 44473000 IC50 = 100 nM T13714 C31XLA 44473001 IC50 = 12 nM T13714 CI7C5U 44473002 IC50 = 3 nM T13714 CFMP64 44473003 IC50 = 6 nM T13714 C01LIU 44473004 IC50 = 7 nM T13714 CR5SI0 44476535 EC50 > 10000 nM T13714 CDY1W2 44537910 IC50 > 30000 nM T13714 C0OC3N 44559230 EC50 > 50000 nM T13714 CW5RK4 44559244 EC50 > 50000 nM T13714 CEYC85 44564595 EC50 = 43 nM T13714 CV9MX0 44568830 IC50 = 15 nM T13714 CK0TW9 44573589 EC50 = 959 nM T13714 CJW4Z1 44573631 EC50 = 626 nM T13714 C2G3FO 44573632 EC50 = 1500 nM T13714 CTOW18 44573633 EC50 = 790 nM T13714 C18HPE 44573634 EC50 = 880 nM T13714 CQ97MR 44573677 EC50 = 940 nM T13714 C3DS6K 44573678 EC50 = 580 nM T13714 CL4G0H 44573679 EC50 = 2320 nM T13714 C89JSN 44573717 EC50 > 30000 nM T13714 C63LBJ 44573718 EC50 = 3500 nM T13714 C2M5UG 44573719 EC50 > 30000 nM T13714 C3YB2D 44626292 EC50 = 11 nM T13714 C4GC8P 45100506 EC50 = 79.43 nM T13714 CA41BS 45270660 IC50 = 20000 nM T13714 C0J3SN 45271480 IC50 = 38000 nM T13714 CR8S4O 45272392 EC50 = 10180 nM T13714 CW79BY 45273240 IC50 = 65000 nM T13714 C3MFY7 45273258 EC50 = 4170 nM T13714 CD9HP7 45481812 IC50 > 30000 nM T13714 CS2UX1 45481813 IC50 > 30000 nM T13714 C3PFR7 45481814 IC50 > 30000 nM T13714 C4YMB1 45481815 IC50 > 30000 nM T13714 CZ8Q5T 45481819 IC50 > 30000 nM T13714 CV21SO 45481820 IC50 = 4300 nM T13714 CJPO37 45481822 IC50 > 30000 nM T13714 C52JWR 45481823 IC50 > 30000 nM T13714 C40FHL 45481824 IC50 > 3000 nM T13714 C47JKF 45481825 IC50 > 3000 nM T13714 C43HEV 45481826 IC50 > 30000 nM T13714 CKT4W8 45481827 IC50 > 30000 nM T13714 C0FZ7X 45481832 IC50 > 30000 nM T13714 CL86HQ 45481833 IC50 > 30000 nM T13714 C9BCY0 45481835 IC50 = 7700 nM T13714 CVZ52U 45481836 IC50 > 30000 nM T13714 C07VHN 45481837 IC50 = 17000 nM T13714 C1EDT6 45481838 IC50 > 30000 nM T13714 CL4XN0 45481843 IC50 > 1000 nM T13714 C4MFG7 45481845 IC50 > 30000 nM T13714 CHSL86 45481846 IC50 > 30000 nM T13714 C0WEA4 45481847 IC50 = 14000 nM T13714 C59QUA 45481848 IC50 > 30000 nM T13714 CTV19K 45481849 IC50 > 30000 nM T13714 C94EIX 45481850 IC50 = 21000 nM T13714 CJ0Z8I 45481851 IC50 > 30000 nM T13714 C0RH7Z 45481853 IC50 > 30000 nM T13714 C7WZ9H 45481854 IC50 > 30000 nM T13714 CFV3R5 45481855 IC50 > 30000 nM T13714 C4ORE2 45481858 IC50 > 30000 nM T13714 C69RLK 45481859 IC50 > 30000 nM T13714 CZE8O5 45481861 IC50 = 7600 nM T13714 C8QNC7 45483602 EC50 = 174 nM T13714 CEF0U7 46186945 IC50 = 18 nM T13714 C4WH5O 46191159 EC50 = 630 nM T13714 CW76XG 46191160 EC50 = 1600 nM T13714 C0M8HC 46202578 IC50 > 1000 nM T13714 C2M9LX 46202579 IC50 > 1000 nM T13714 CY0B3G 46202580 IC50 > 1000 nM T13714 CPUM13 46202603 IC50 = 3162.28 nM T13714 CIP60A 46202604 IC50 > 10000 nM T13714 C35THS 46202902 IC50 > 1000 nM T13714 CA41NL 46202903 IC50 = 132 nM T13714 C1HP7B 46202904 IC50 = 81 nM T13714 C6IGM9 46202905 IC50 > 1000 nM T13714 C5LOI9 46202906 IC50 > 1000 nM T13714 CG2K7B 46202907 IC50 = 34 nM T13714 C3NVR5 46202928 IC50 > 10000 nM T13714 CS12DL 46202929 EC50 = 3.162 nM T13714 CVKU68 46202930 EC50 = 1 nM T13714 C0GOL4 46202931 EC50 = 19.95 nM T13714 CF5D2Q 46202932 EC50 = 3.162 nM T13714 CV91AT 46203225 IC50 = 299 nM T13714 C6I3NU 46203226 IC50 = 395 nM T13714 CY34FM 46203248 EC50 = 15.85 nM T13714 CGF3P7 46203249 EC50 = 100 nM T13714 CD0K4Y 46206336 EC50 = 580 nM T13714 C18TZO 46225114 IC50 = 367 nM T13714 CQW01V 46225115 IC50 = 730 nM T13714 C4VBQ8 46225151 IC50 = 5294 nM T13714 C1M2NC 46225152 IC50 = 77 nM T13714 CB94AX 46225194 IC50 = 5133 nM T13714 CZL91B 46225195 IC50 = 18 nM T13714 C8P3HN 46225196 IC50 = 62 nM T13714 CZ7K6G 46225197 IC50 = 11 nM T13714 C9FD3L 46225243 IC50 = 57 nM T13714 CQ94OV 46225244 IC50 = 5 nM T13714 C2R5PZ 46225245 IC50 = 28 nM T13714 CO56AF 46225246 IC50 = 590 nM T13714 CE2W0C 46225296 IC50 = 2850 nM T13714 CN9JT0 46226318 EC50 = 4100 nM T13714 CT3E5K 46226367 IC50 > 1000 nM T13714 C4KVS8 46226434 IC50 > 1000 nM T13714 C4NM1R 46226975 IC50 = 129 nM T13714 C1JA3L 46838908 Ki = 99000 nM T13714 CR6X9K 46877573 EC50 = 1860 nM T13714 C4QTV3 46877575 IC50 > 1000 nM T13714 C9LQM2 46877576 EC50 = 920 nM T13714 C9DVO7 46877577 EC50 = 170 nM T13714 C0YDO7 46877578 EC50 = 1700 nM T13714 CN0VI5 46886359 IC50 = 398.11 nM T13714 COJN09 46887743 IC50 > 1000 nM T13714 C0Q8VO 46887744 EC50 = 284 nM T13714 CJW63M 46887745 IC50 = 355 nM T13714 C0PK3A 46887797 EC50 = 100 nM T13714 CQCD45 46887798 IC50 = 109 nM T13714 CM23GQ 46887799 IC50 = 2.4 nM T13714 CCG9X7 46887800 EC50 = 106 nM T13714 CK41YM 46887851 EC50 = 91 nM T13714 CFY72K 46887852 EC50 = 1080 nM T13714 CDPU51 46887853 EC50 = 580 nM T13714 C1D6VN 46887854 EC50 = 175 nM T13714 C3ZMN8 46887888 IC50 = 629 nM T13714 C8BLU0 46887889 EC50 = 161 nM T13714 COL94T 46887890 EC50 = 195 nM T13714 CYI8F3 46887891 EC50 = 512 nM T13714 CVX9L5 46887924 EC50 = 565 nM T13714 CN9L7G 46916268 EC50 > 8300 nM T13714 CP56CJ 49821979 EC50 = 12 nM T13714 C3HQK9 49821981 EC50 = 2 nM T13714 C4LZ1T 49822063 EC50 = 2 nM T13714 CPT4Z8 49822066 EC50 = 5 nM T13714 CIJ50V 49822147 EC50 = 2 nM T13714 CMPO56 49822148 EC50 = 3 nM T13714 CG6LI3 49822225 EC50 = 8 nM T13714 C5CG6O 49822226 EC50 = 1 nM T13714 CUD91T 49862248 EC50 > 10000 nM T13714 CL78UE 54344821 EC50 = 3040 nM T13714 C5ZX4B 54597874 IC50 > 10000 nM T13714 CUT56J 56589730 EC50 = 1150 nM T13714 C7DQ1X 57404459 IC50 = 800 nM T13714 CFVN93 57757122 EC50 = 100 nM T13714 C4BTN7 57900760 EC50 = 1000 nM T13714 C9XA5G 57900823 EC50 = 860 nM T13714 CVW8C9 57962776 EC50 = 8000 nM T13714 CENS58 57962786 EC50 = 1000 nM T13714 CCU2Q0 57962869 EC50 = 2400 nM T13714 CU1D2E 57962891 EC50 = 960 nM T13714 CF79JZ 57962903 EC50 = 2000 nM T13714 C1SJN3 57962913 EC50 = 1400 nM T13714 C9PD2F 57962932 EC50 = 1300 nM T13714 C63ZOK 57962935 EC50 = 1300 nM T13714 CB16MY 57962948 EC50 = 3000 nM T13714 C6Q5TV 57962956 EC50 = 4700 nM T13714 COZ0J7 57962965 EC50 = 1300 nM T13714 CJE7R4 57962994 EC50 = 5300 nM T13714 C8CY6K 57963018 EC50 = 1300 nM T13714 CKH02U 59200932 EC50 = 1880 nM T13714 CI6O2P 59200935 EC50 = 2870 nM T13714 CU6Z4C 59200977 EC50 = 700 nM T13714 C9VZN3 59200986 EC50 = 2850 nM T13714 C5F7IQ 59201030 EC50 = 1660 nM T13714 C2HYE6 59201075 EC50 = 500 nM T13714 C0OD8R 59201087 EC50 = 110 nM T13714 C23OUL 59201095 EC50 = 1810 nM T13714 CRJ3Q2 59201115 EC50 = 7 nM T13714 C8EB3H 59201131 EC50 = 120 nM T13714 CHLR48 59234874 EC50 = 1200 nM T13714 C73CIF 59234887 EC50 = 1700 nM T13714 CH78VI 59234921 EC50 = 700 nM T13714 CIB7H4 59234952 EC50 = 1300 nM T13714 CE9J7G 59234955 EC50 = 1000 nM T13714 CT8QH0 59234958 EC50 = 600 nM T13714 CSF58L 59234986 EC50 = 610 nM T13714 C2B4OJ 59234998 EC50 = 1100 nM T13714 C2YS3R 59234999 EC50 = 2700 nM T13714 C8E3TC 59235012 EC50 = 560 nM T13714 C6R0AK 59235049 EC50 = 1300 nM T13714 C7F5KX 59235054 EC50 = 700 nM T13714 CJUK93 59235080 EC50 = 400 nM T13714 C1E4JW 59235082 EC50 = 800 nM T13714 C84TQU 59235084 EC50 = 1100 nM T13714 CK1JR4 59235110 EC50 = 1000 nM T13714 CK08IO 59235130 EC50 = 100 nM T13714 C3QE7W 59235136 EC50 = 1600 nM T13714 CTO4C0 59235143 EC50 = 1400 nM T13714 CEQD45 59235170 EC50 = 700 nM T13714 C92RGU 59251295 EC50 = 61 nM T13714 CES06G 59251431 EC50 = 670 nM T13714 CG2NL0 59251456 EC50 = 140 nM T13714 CU02IZ 59251553 EC50 = 66 nM T13714 C17SAE 59251574 EC50 = 9 nM T13714 C17AXL 59251592 EC50 = 600 nM T13714 C36TYG 59631866 EC50 = 620 nM T13714 C4LTZ9 59631939 EC50 = 64 nM T13714 CN15OH 59632480 EC50 = 49 nM T13714 CE1K9L 59632482 EC50 = 108 nM T13714 CUVR29 59632565 EC50 = 68 nM T13714 CAKQ02 59633156 EC50 = 230 nM T13714 CJ36PA 59726531 EC50 = 2 nM T13714 CKO07V 61343280 EC50 = 68 nM T13714 CPAB97 61352587 EC50 = 493 nM T13714 CD76EJ 61353182 EC50 = 68 nM T13714 C5H6NQ 66797441 EC50 = 320 nM T13714 CS41OX 67119337 EC50 = 530 nM T13714 CAD80C 68469431 Ki = 35000 nM T13714 CP1M5T 68655604 EC50 = 14 nM T13714 C1B7QU 70682541 IC50 = 160 nM T13714 CM9WS7 70682542 IC50 > 10000 nM T13714 C42MZQ 70682550 IC50 = 300 nM T13714 C69XGS 70684628 IC50 = 700 nM T13714 C7CD6G 70684639 IC50 = 500 nM T13714 CY5C0F 70686771 IC50 > 10000 nM T13714 CS2K3Z 70686772 IC50 = 3600 nM T13714 CYG6W5 70686773 IC50 > 10000 nM T13714 C15QVE 70686781 IC50 = 600 nM T13714 C39IFO 70686782 IC50 = 1200 nM T13714 CQ9SP8 70686783 IC50 = 150 nM T13714 CC8A4N 70688856 IC50 = 1100 nM T13714 C35QCK 70688857 IC50 = 5100 nM T13714 CF45TP 70688865 IC50 > 10000 nM T13714 C32AVT 70688866 IC50 = 1800 nM T13714 CS0X2G 70690946 IC50 = 400 nM T13714 CS43WF 70690947 IC50 = 1000 nM T13714 CNA0I1 70693085 IC50 = 3200 nM T13714 CN9SV5 70693093 IC50 = 4300 nM T13714 CRK50F 70693094 IC50 = 10000 nM T13714 C3C2FA 70695131 IC50 = 1500 nM T13714 CT8CN0 70695140 IC50 = 3500 nM T13714 CG3F1Z 70697168 IC50 > 10000 nM T13714 CC3M6V 70697169 IC50 = 1000 nM T13714 CM0E8T 70697178 IC50 = 10000 nM T13714 CH3P1A 70697179 IC50 = 600 nM T13714 C5B7DK 71451721 IC50 = 15000 nM T13714 C4WVB2 71451730 IC50 > 10000 nM T13714 C2J0LM 71451731 IC50 > 10000 nM T13714 CM6Z3K 71455271 EC50 = 2700 nM T13714 CGJ60X 71455272 IC50 > 30000 nM T13714 CGE0M4 71457060 IC50 = 27000 nM T13714 CEO4U2 71457061 IC50 = 7500 nM T13714 CTY76D 71457062 EC50 = 260 nM T13714 CP50ZQ 71458918 IC50 = 11000 nM T13714 C3YL4V 71458919 IC50 = 26000 nM T13714 CDM21R 71460722 IC50 = 9500 nM T13714 C8UKI7 71460723 IC50 = 27000 nM T13714 CQU5I1 71460728 IC50 > 30000 nM T13714 C1C3OQ 71460729 IC50 > 30000 nM T13714 C8JXP0 71462452 IC50 = 13000 nM T13714 C9Z2MA 71462453 IC50 > 10000 nM T13714 CPS62O 71462454 EC50 = 770 nM T13714 CZ9E2O 71462455 IC50 > 10000 nM T13714 CT47LS 71462456 IC50 > 10000 nM T13714 C1DR8E 71622396 EC50 = 2500 nM T13714 CKV30T 72207455 Ki = 16000 nM T13714 C4KZ9W 72529513 EC50 = 64 nM T13714 CMZ85K 72722807 EC50 = 902 nM T13714 C2BQO3 72722945 EC50 = 385 nM T13714 C6UWO5 74762670 EC50 > 10000 nM T13714 CJXG25 76284182 EC50 > 10000 nM T13714 CMW6O1 77620538 EC50 = 3900 nM T13714 C7ZMD9 78319220 IC50 = 680 nM T13714 CV64IH 86233643 EC50 = 259 nM T13714 C7ZM1B 86297437 EC50 = 40 nM T13714 C4SA8H 86302482 EC50 > 10000 nM T13714 CBI06J 86346645 EC50 > 10000 nM T13714 C5VCM4 86690644 EC50 > 10000 nM T13714 CGFW70 86690646 EC50 > 10000 nM T13714 C5J9MZ 87123143 EC50 = 800 nM T13714 CGA6W0 87123160 EC50 = 12000 nM T13714 CB4Y0Z 87198339 EC50 = 360 nM T13714 C5MOV2 89659415 EC50 > 10000 nM T13714 CLW3O5 89665055 EC50 = 3800 nM T13714 C7E5RV 90200534 EC50 > 10000 nM T13714 C15KAB 90447258 EC50 = 110 nM T13714 CA2LF3 90447465 EC50 = 651 nM T13714 CUS5A8 90447547 EC50 = 16 nM T13714 CS53WO 91663364 EC50 = 560 nM T13714 CG0N9Y 91663938 Ki = 209000 nM T13714 CI92WR 91664317 EC50 > 10000 nM T13714 CU96JS 91800925 Ki = 18000 nM T13714 CI0J1E 91827511 EC50 = 210 nM T13714 CT3K8B 117940657 EC50 > 7500 nM T13714 C9R5HF 117949985 EC50 > 7500 nM T13714 C0W6MZ 117950226 EC50 = 3710 nM T13714 C39DHO 117951324 EC50 = 18 nM T13714 C4S9EM 117964962 EC50 > 10000 nM T13714 CS4GJ9 117964973 EC50 > 10000 nM T13714 CDXK37 117964975 EC50 > 10000 nM T13714 CN6RT8 117964978 EC50 > 10000 nM T13714 C96BSK 117964998 EC50 > 10000 nM T13714 C79IOD 118207841 EC50 > 7500 nM T13714 CW27ZE 118207854 EC50 > 7500 nM T13714 C2FLM1 118207907 EC50 > 7500 nM T13714 CXW5M0 118207954 EC50 > 7500 nM T13714 C9UK5A 118207966 EC50 > 7500 nM T13714 C0SQH5 118207970 EC50 > 7500 nM T13714 C0PWH6 118207991 EC50 > 7500 nM T13714 C2U3TJ 118208018 EC50 > 7500 nM T13714 C1MOT7 118208026 EC50 > 7500 nM T13714 CZ2C3U 118208048 EC50 > 7500 nM T13714 CI86YW 118208079 EC50 > 7500 nM T13714 C2KAR6 118208086 EC50 > 7500 nM T13714 C3TJY2 118208092 EC50 > 7500 nM T13714 CS2F1K 118208112 EC50 > 7500 nM T13714 C8N2PF 118208184 EC50 > 7500 nM T13714 C51XTL 118217548 EC50 > 7500 nM T13714 C1FL5I 118217550 EC50 > 7500 nM T13714 CEN76C 118217555 EC50 > 7500 nM T13714 CYRF01 118217561 EC50 = 1900 nM T13714 C2LIW9 118217576 EC50 > 7500 nM T13714 CH9T1O 118217580 EC50 > 7500 nM T13714 CIT31Q 118217593 EC50 > 7500 nM T13714 C1ZRN9 118217594 EC50 > 7500 nM T13714 CAUT58 118217595 EC50 > 7500 nM T13714 CB3KO0 118217596 EC50 > 7500 nM T13714 C95ERM 118217608 EC50 > 7500 nM T13714 CM2U4C 118217609 EC50 > 7500 nM T13714 C9V0ZM 118217611 EC50 > 7500 nM T13714 CZ5L3N 118217612 EC50 > 7500 nM T13714 CCK3J9 118217851 EC50 > 7500 nM T13714 CO5I3V 118217852 EC50 > 7500 nM T13714 CD5TJ3 118217853 EC50 > 7500 nM T13714 C6HSC3 118217854 EC50 > 7500 nM T13714 CEKH57 118217858 EC50 > 7500 nM T13714 C1CTB6 118217859 EC50 > 7500 nM T13714 C7U0XR 118217863 EC50 > 7500 nM T13714 CDP0H5 118217865 EC50 > 7500 nM T13714 C82YDU 118217866 EC50 > 7500 nM T13714 CQ60HK 118217867 EC50 > 7500 nM T13714 C9N7VY 118217868 EC50 > 7500 nM T13714 C6LC7H 118217869 EC50 > 7500 nM T13714 CV9G4S 118217870 EC50 > 7500 nM T13714 C8PR3G 118217871 EC50 > 7500 nM T13714 CZ3FX6 118217874 EC50 > 7500 nM T13714 CK85HV 118217875 EC50 > 7500 nM T13714 CT0DV4 118217911 EC50 > 7500 nM T13714 C1QPW5 118217915 EC50 > 7500 nM T13714 C3YTM2 118217920 EC50 > 7500 nM T13714 CU0T7K 118217922 EC50 > 7500 nM T13714 C0ETA2 118217925 EC50 > 7500 nM T13714 C89EDG 118217927 EC50 > 7500 nM T13714 C81QMJ 118217932 EC50 > 7500 nM T13714 C6X4IN 118217935 EC50 > 7500 nM T13714 CD01CA 118526849 EC50 > 10000 nM T13714 CBZ75K 118724654 EC50 > 10000 nM T13714 CAT4B6 118729956 EC50 = 1400 nM T13714 CSX13I 118729957 EC50 = 2200 nM T13714 CU08LA 118796406 EC50 = 2310 nM T13714 CQNI87 118883423 Ki = 1 nM T13714 CP75LI 118883429 Ki = 9 nM T13714 CB6F8J 118883492 Ki = 8 nM T13714 CY29BV 118987028 EC50 = 30 nM T13714 C3RFZ1 121596966 Ki = 6 nM T13714 CP52DJ 121596967 Ki = 13 nM T13714 CYJX02 122180565 EC50 = 2000 nM T13714 CWV50E 122181445 EC50 = 2200 nM T13714 CRY8N5 122190169 EC50 = 5700 nM T13714 C9QF1B 122192262 IC50 > 30000 nM T13714 C34OXY 122192263 IC50 > 30000 nM T13714 CE76CW 122192264 IC50 > 30000 nM T13714 CN0D3U 122192265 IC50 > 30000 nM T13714 C3C2MX 122192266 IC50 > 30000 nM T13714 CSHD20 122192267 IC50 > 30000 nM T13714 CHDI48 122192268 IC50 > 30000 nM T13714 CF5Q8I 122192269 IC50 > 30000 nM T13714 C6MEU5 122192270 IC50 = 6800 nM T13714 C58SCX 122192271 IC50 > 30000 nM T13714 C53ACS 122192272 IC50 > 30000 nM T13714 CLJ7S1 122192273 IC50 = 1800 nM T13714 C4UO8G 122192274 IC50 = 15000 nM T13714 CZ6X9G 122192275 IC50 > 30000 nM T13714 CPI25Z 122192276 IC50 = 21000 nM T13714 C8E9GN 122192277 IC50 = 25000 nM T13714 CJ30NY 122192278 IC50 > 30000 nM T13714 C80QHL 122192280 IC50 > 30000 nM T13714 C4F9ZK 122669103 IC50 > 10000 nM T13714 CZH39M 122669106 IC50 > 10000 nM T13714 C0T8FO 122669173 IC50 > 10000 nM T13714 CD6X5P 122669265 EC50 > 7500 nM T13714 C0S7UB 122678562 IC50 > 10000 nM T13714 CY8S1P 122678563 IC50 > 10000 nM T13714 C0MUW2 122678576 IC50 > 10000 nM T13714 C2SQ9M 122678748 IC50 > 10000 nM T13714 CH1J6K 122678779 IC50 > 10000 nM T13714 CD9HN3 122678983 IC50 > 10000 nM T13714 CF39TE 122679031 IC50 > 10000 nM T13714 CW37BU 127044455 EC50 = 770 nM T13714 CYO9Q7 127044456 EC50 = 7 nM T13714 C1L5VC 127044605 EC50 = 550 nM T13714 C9QO3M 127044780 EC50 = 840 nM T13714 CW46GA 127049311 EC50 > 20000 nM T13714 CZW30P 127049312 Ki = 94 nM T13714 CKM23U 127049313 Ki = 4 nM T13714 CB1IR7 127051155 Ki = 460 nM T13714 C1RC3J 127052439 EC50 = 2330 nM T13714 C8JW1U 129167185 EC50 = 223 nM T13714 CB62QX 131953519 EC50 > 7500 nM T13714 CK0G6A 134131424 Ki = 26 nM T13714 CES87G 134135247 Ki = 1 nM T13714 C2A7CZ 134138904 Ki = 13 nM T13714 CBSF46 134142531 EC50 = 12 nM T13714 C8MAB7 134142736 Ki = 13 nM T13714 CVC1Y4 134142943 Ki = 4 nM T13714 CK13YN 134145788 Ki = 5 nM T13714 CR0OX5 134146533 EC50 = 8 nM T13714 CB39QU 134150059 EC50 = 21 nM T13714 C9NI7K 134151534 Ki = 6 nM T13714 CZH50T 134151855 Ki = 6 nM T13714 C0LGI2 134154676 Ki = 7 nM T13714 CZV9B3 134154775 Ki = 7 nM T13714 CJ0UG1 134155310 EC50 = 16 nM T13714 CNS38M 134157776 Ki = 3 nM T13714 CW9Y7T 135410235 EC50 = 19000 nM T13714 C1DTF0 137634167 EC50 = 2700 nM T13714 C7R8XI 137635446 EC50 = 12720 nM T13714 CN40KU 137638307 EC50 = 1960 nM T13714 C6PSI1 137641894 EC50 = 3790 nM T13714 C5W2UL 137643175 EC50 = 1960 nM T13714 CE21KT 137651926 EC50 = 6020 nM T13714 CXQ9V8 137659428 EC50 = 7200 nM T13714 CK3X1N 137796283 EC50 > 30000 nM T13714 CC2BH9 145232219 EC50 > 30000 nM T13714 CW3Y0H 145949340 IC50 > 20000 nM T13714 CPK5U1 145951022 IC50 > 20000 nM T13714 CZM2D7 145963820 EC50 = 130 nM T13714 CI3TP7 145964673 EC50 = 2470 nM T13714 CE01FB 145964868 EC50 = 8000 nM T13714 CFK0H4 145965098 EC50 = 340 nM T13714 CX6T7R 145965139 EC50 = 4960 nM T13714 CKL63D 145965344 EC50 > 7500 nM T13714 C3GI6D 145965669 EC50 > 7500 nM T13714 C4TL7G 145965870 EC50 = 2900 nM T13714 C4H9UY 145966156 EC50 = 185 nM T13714 C3B8PL 145966450 EC50 = 8980 nM T13714 C4P3DR 145967002 EC50 = 2820 nM T13714 C8C4GB 145967545 EC50 > 10000 nM T13714 CY1X5Q 145968478 EC50 > 7500 nM T13714 CG27VL 145969403 EC50 = 1040 nM T13714 CYT8M9 145971562 EC50 > 7500 nM T13714 C3WZG1 145972771 EC50 = 4670 nM T13714 CN3U9C 145973265 EC50 = 4770 nM T13714 CC8HN9 145973516 EC50 = 3120 nM T13714 CYA1D0 145973564 EC50 = 915 nM T13714 C0X3EB 145974156 EC50 > 7500 nM T13714 C3UI5R 145974164 EC50 = 270 nM T13714 C13TQJ 145974494 EC50 = 455 nM T13714 CAYQ72 145974767 EC50 = 370 nM T13714 C4SPY0 145974975 EC50 = 559 nM T13714 C47KPT 145975021 EC50 > 10000 nM T13714 C37NDQ 145975104 EC50 = 3610 nM T13714 C60CDE 145975835 EC50 > 7500 nM T13714 CA3XR1 145976113 EC50 = 2450 nM T13714 CQZ7I9 145977465 EC50 = 445 nM T13714 CE2O1P 145977892 EC50 = 550 nM T13714 CB70AE 145980094 EC50 > 30000 nM T13714 CRTG03 145987785 EC50 > 30000 nM T13714 CO8R4D 145989300 EC50 = 720 nM T13714 CC89OI 148034311 IC50 > 10000 nM T13714 CE6V8Z 155511797 IC50 > 10000 nM T13714 C9D7ZE 155515113 EC50 = 1425 nM T13714 C14OPD 155516918 EC50 = 966 nM T13714 C6SBY9 155521216 EC50 = 109 nM T13714 CU5Z8T 155522788 IC50 > 10000 nM T13714 C1DT9M 155525669 IC50 > 10000 nM T13714 CXS9T8 155526989 IC50 > 10000 nM T13714 C59SQP 155528665 EC50 = 2365 nM T13714 C35CIV 155530360 Ki = 7342 nM T13714 CO9N5H 155530678 IC50 > 10000 nM T13714 CIUA10 155537856 IC50 > 10000 nM T13714 CLO98T 155539150 EC50 > 7500 nM T13714 CDU60J 155539858 EC50 = 712 nM T13714 CY4OQ3 155541483 EC50 = 5647 nM T13714 C0V6EY 155543172 IC50 > 10000 nM T13714 CX7L0S 155544387 IC50 > 10000 nM T13714 CSK20E 155544524 IC50 > 10000 nM T13714 CTEC81 155544796 EC50 > 7500 nM T13714 CBK1E5 155556708 IC50 > 10000 nM T13714 CH62VW 155557200 EC50 = 6706 nM T13714 C3FI7U 155560819 IC50 > 10000 nM T13714 CA91EM 155564933 IC50 > 10000 nM T13714 CPF42S 155565257 IC50 > 10000 nM T13714 C1AJO9 155568648 EC50 = 231 nM T13714 D00DLU 16049480 IC50 = 30 nM T13714 D00HVP 10070992 IC50 = 6600 nM T13714 D02UID 16734800 Ki = 14.2 nM T13714 D06VRA 24860515 IC50 = 7300 nM T13714 D07XLQ 44537911 IC50 > 30000 nM T13714 D08QXD 9935197 EC50 = 16 nM T13714 D09UND 24860514 IC50 = 14000 nM T13714 D09VLE 24860516 IC50 = 77000 nM T13714 D0A1WR 71478195 IC50 = 43 nM T13714 D0B5FC 447912 EC50 = 4.7 nM T13714 D0C6QI 9830426 EC50 < 3 nM T13714 D0HA0U 24860512 IC50 = 7600 nM T13714 D0IZ9O 24860513 IC50 = 10000 nM T13714 D0K4GK 167685 EC50 = 4750 nM T13714 D0L1CX 45481863 IC50 > 30000 nM T13714 D0PL4F 447905 Ki = 2.2 nM T13714 D0Q2RP 3247059 EC50 = 168 nM T13714 D0R8LN 45481844 IC50 = 3500 nM T13714 D0U4TN 10638446 IC50 = 65000 nM T13714 D0V3PG 128861 EC50 = 125200 nM T13714 D0V4RZ 25113722 IC50 = 33 nM T13714 D0X2HK 45481821 IC50 > 30000 nM T13714 D0X5DT 10616182 IC50 > 30000 nM T13714 D0Z3TJ 46203250 IC50 = 31.62 nM T13714 D0Z8LE 24860511 IC50 = 13000 nM T13714 D0Z8RH 25137977 IC50 = 41 nM T47107 D09DHT 27924 Ki = 4.9 nM T47107 D0E3TC 44259 IC50 = 2.76 nM T47107 D0I6VU 176167 IC50 = 83 nM T47107 D0S5RC 3025986 IC50 > 40000 nM T47107 D0W3LI 153999 IC50 = 300 nM T47107 D03BNU 59604787 IC50 > 10000 nM T47107 D0WS1V 448991 IC50 > 100000 nM T47107 D0R2TM 5287736 IC50 = 10 nM T47107 D0T3ME 156422 IC50 > 30000 nM T47107 C8OI7N 2290 IC50 = 30 nM T47107 C95GCZ 3568 IC50 = 50000 nM T47107 CJ17AM 4877 IC50 > 100000 nM T47107 CG2P1X 159320 Ki = 1.2 nM T47107 C8PU1O 188534 Ki = 15 nM T47107 CMN15U 192686 IC50 = 34000 nM T47107 C0G6JH 455733 Ki = 3100 nM T47107 C6DLK3 644364 IC50 = 2700 nM T47107 CLA43B 5327919 IC50 = 60 nM T47107 CPDC54 5327920 IC50 = 2200 nM T47107 CCB9G3 5327921 IC50 = 13 nM T47107 CRTQ98 5327922 IC50 = 10 nM T47107 CP20NQ 5327923 IC50 = 35 nM T47107 C98CNM 5327943 IC50 = 6600 nM T47107 C61URB 5327944 IC50 = 10 nM T47107 CWUY53 5327945 IC50 = 3500 nM T47107 CQ54BE 5327946 IC50 = 220 nM T47107 CIB3P0 5327947 IC50 = 2600 nM T47107 CVG0A1 5327948 IC50 = 470 nM T47107 C8M3PD 5327949 IC50 = 5000 nM T47107 COP0Q2 5327951 IC50 = 4200 nM T47107 CB47VN 5327952 IC50 = 830 nM T47107 CPO51K 5327953 IC50 = 250 nM T47107 CI6AY9 5327954 IC50 = 2900 nM T47107 C1Q0PM 5327955 IC50 = 4800 nM T47107 CXA23M 5327956 IC50 = 1600 nM T47107 CH73DT 5327957 IC50 = 1400 nM T47107 CTI6K8 5327963 IC50 = 4100 nM T47107 CAO1N9 5327979 IC50 = 1100 nM T47107 CZ3LK2 5330387 IC50 > 10000 nM T47107 C2RA4O 5352033 Ki = 0.38 nM T47107 CG17TN 6914611 IC50 = 270 nM T47107 C7E2QK 6914613 IC50 = 1200 nM T47107 CBT0X5 9797847 IC50 = 56500 nM T47107 C4PA5X 9800852 Ki = 279 nM T47107 C8J1OL 9826373 IC50 = 400 nM T47107 CCJK12 9865633 Ki = 40.7 nM T47107 C20NKA 9889351 IC50 = 500 nM T47107 CQD2W7 9935079 IC50 = 1200 nM T47107 CP5NJ3 9952970 Ki = 140 nM T47107 CV34AB 9958125 IC50 = 7000 nM T47107 CJ84TX 9977154 IC50 = 5500 nM T47107 C2W3AV 9995236 IC50 = 2000 nM T47107 C57DLH 10001523 IC50 = 3600 nM T47107 CV7Z9Y 10002471 IC50 = 2800 nM T47107 C2UGV9 10030483 IC50 = 1000 nM T47107 CO5KL3 10072710 IC50 = 6000 nM T47107 CT6BJ7 10099352 IC50 = 74000 nM T47107 CG7JO8 10099482 IC50 = 1000 nM T47107 C93LPQ 10099652 IC50 = 140 nM T47107 CFXZ38 10114332 IC50 > 10000 nM T47107 CRT67V 10119173 IC50 = 1570 nM T47107 CZJI60 10141037 IC50 > 10000 nM T47107 C94WRY 10143231 IC50 > 10000 nM T47107 C76TVG 10143584 IC50 = 3400 nM T47107 CY7W1Z 10144680 IC50 = 5170 nM T47107 CLBD08 10144909 IC50 = 340 nM T47107 C7JP1A 10163439 IC50 = 210 nM T47107 C3QZV8 10184859 IC50 = 370 nM T47107 CJN72C 10185160 IC50 = 280 nM T47107 CJ0R2G 10187378 IC50 = 710 nM T47107 C73LXY 10188021 IC50 = 510 nM T47107 CK7UT9 10188786 IC50 = 1300 nM T47107 C5P8JC 10206423 IC50 = 1340 nM T47107 CGOT91 10207821 IC50 = 300 nM T47107 CUF0W9 10207822 IC50 = 980 nM T47107 C98TUI 10208507 IC50 = 400 nM T47107 C0IYO3 10208648 IC50 = 3300 nM T47107 C51SKM 10209082 IC50 = 110 nM T47107 CK72XG 10209108 IC50 = 250 nM T47107 CI8MW4 10216627 IC50 = 540 nM T47107 C3VK7T 10229967 IC50 = 1570 nM T47107 C2X6LY 10275064 IC50 = 2730 nM T47107 C7U9BE 10281603 IC50 > 10000 nM T47107 CTXN56 10296960 IC50 = 320 nM T47107 C4F1YI 10297128 IC50 = 2670 nM T47107 CAX9W2 10302405 IC50 = 47 nM T47107 CHB84X 10341165 IC50 = 8700 nM T47107 CFU38G 10363814 Ki = 2820 nM T47107 CEH41V 10392789 IC50 = 5 nM T47107 C3RBY8 10395226 Ki > 500 nM T47107 CRVE78 10411641 IC50 = 8600 nM T47107 CQXJ51 10425978 Ki = 288.1 nM T47107 C36QRS 10453829 Ki = 970 nM T47107 C10PAC 10460251 IC50 = 5 nM T47107 C25LDK 10460643 IC50 = 32000 nM T47107 CMA4J8 10479260 Ki = 327 nM T47107 CX7S8N 10482293 IC50 = 5 nM T47107 C76QGP 10506540 IC50 = 30 nM T47107 CSR8Y5 10527068 IC50 = 2100 nM T47107 CDNP37 10530708 IC50 = 50 nM T47107 C5EYJ3 10554684 IC50 = 400 nM T47107 C71UIS 10555532 IC50 = 4300 nM T47107 CZ8UA9 10650891 IC50 > 5000 nM T47107 CJOU71 10671412 IC50 = 270 nM T47107 CM5B6A 10673286 IC50 = 2500 nM T47107 CN9I6T 10768377 IC50 = 3200 nM T47107 CL8VH3 10768554 IC50 = 6500 nM T47107 C5YMK8 10769011 IC50 = 10 nM T47107 C7HPA0 10864309 IC50 = 5000 nM T47107 C1DRE5 10884145 IC50 > 150 ug.mL-1 T47107 C2G5CU 10894726 Ki = 6320 nM T47107 C1L4ZC 10940039 IC50 = 3500 nM T47107 CR47CD 11025838 Ki = 675 nM T47107 CBOP58 11293798 Ki > 10000 nM T47107 C26BZX 11362471 Ki > 10000 nM T47107 CWXB93 11397177 Ki > 10000 nM T47107 C8DNQ2 11453012 IC50 = 2000 nM T47107 CTG83F 11539329 Ki > 8800 nM T47107 CACS26 11561968 Ki > 10000 nM T47107 CMIL86 11590363 Ki > 8800 nM T47107 C9T6SC 11640926 Ki > 8800 nM T47107 CU0E8O 11690457 Ki = 210 nM T47107 CB0AP2 11705863 Ki > 4000 nM T47107 CCX53Q 11729563 IC50 = 500 nM T47107 CM10YB 11799388 IC50 = 2200 nM T47107 CA05OS 11972484 IC50 = 210 nM T47107 C2BX8F 15297223 IC50 = 300 nM T47107 CE04YW 15297224 IC50 = 46000 nM T47107 C7N6CQ 15604547 IC50 = 31 nM T47107 CFPW41 16007116 Ki > 8800 nM T47107 C9TU1O 16046126 IC50 > 1000 nM T47107 CC24KI 16667248 IC50 = 1560 nM T47107 CS15LY 21672114 Ki = 0.63 nM T47107 CVR9K4 22907281 IC50 = 1300 nM T47107 C0HRM6 22911602 IC50 = 300 nM T47107 CUN67H 23366085 IC50 = 170 nM T47107 CLG9Z8 23366090 IC50 = 4600 nM T47107 CKYB29 23644745 IC50 = 50 nM T47107 C2JTA3 23647573 IC50 = 260 nM T47107 CK73JS 24742033 Ki = 420 nM T47107 CX1HL8 25032704 Ki > 8750 nM T47107 CD5Z8U 44139091 Ki = 35 nM T47107 CAI56R 44139212 Ki = 50.8 nM T47107 CNX5R1 44139336 Ki = 12.3 nM T47107 CRD90G 44139337 Ki = 6.2 nM T47107 C4UMB7 44158300 Ki = 39 nM T47107 C4G5DI 44158301 Ki = 1600 nM T47107 CQ13XB 44291629 Ki > 500 nM T47107 CERT91 44291669 Ki > 500 nM T47107 C1FZ6B 44294270 IC50 = 1700 nM T47107 C6A9FK 44294365 IC50 = 12 nM T47107 C4HS3C 44294447 IC50 = 40 nM T47107 CFZ31C 44294493 IC50 = 250 nM T47107 C54GFD 44294623 IC50 = 5 nM T47107 CG89DS 44294661 IC50 = 380 nM T47107 CG1Z2B 44303442 IC50 = 40 nM T47107 CNJ63O 44303517 IC50 = 330 nM T47107 C8RJN7 44303745 IC50 = 420 nM T47107 CTM59P 44308069 IC50 = 5 nM T47107 CJ4WB9 44308383 IC50 = 30 nM T47107 C1N6SL 44308409 IC50 = 1000 nM T47107 CO83HF 44308467 IC50 = 1000 nM T47107 CYTA85 44308468 IC50 = 4300 nM T47107 C3M4UP 44308469 IC50 = 60 nM T47107 CY4K5F 44308490 IC50 = 34 nM T47107 C7AG9Y 44308609 IC50 = 5 nM T47107 CYN34A 44308610 IC50 = 10 nM T47107 C79WUE 44308611 IC50 = 5 nM T47107 CS63CK 44308612 IC50 = 45 nM T47107 C47BNR 44310732 IC50 = 34 nM T47107 C2ACB1 44310758 IC50 = 10 nM T47107 CXVB19 44310795 IC50 = 1600 nM T47107 CD8OF2 44311036 IC50 = 14 nM T47107 C13TNU 44315122 IC50 = 260 nM T47107 C3YN1R 44315123 IC50 = 390 nM T47107 CPJ57U 44315124 IC50 = 90 nM T47107 C9HA8T 44315171 IC50 = 20 nM T47107 C2T3VN 44315184 IC50 = 210 nM T47107 C3SP0H 44315423 IC50 = 410 nM T47107 C8OAE9 44315457 IC50 = 400 nM T47107 C3JS6X 44315503 IC50 = 40 nM T47107 CEZ68T 44315545 IC50 = 540 nM T47107 CF61IT 44334334 IC50 = 390 nM T47107 C3BFI4 44334443 IC50 = 1000 nM T47107 COJ73E 44355185 Ki = 1.5 nM T47107 CIH03D 44366053 IC50 = 4500 nM T47107 CO28BT 44376126 Ki = 1.84 nM T47107 C8X0WA 44384580 Ki = 209 nM T47107 CC95JU 44385548 IC50 = 400 nM T47107 CGQ57L 44386180 IC50 < 30 nM T47107 CI0Y5L 44386181 IC50 = 10 nM T47107 C1W6NC 44386587 IC50 = 12 nM T47107 C0PU3I 44386588 IC50 = 160 nM T47107 C3J6ZO 44386589 IC50 = 50 nM T47107 C4MZI9 44386931 IC50 = 34000 nM T47107 CETQ79 44427518 IC50 > 50000 nM T47107 COPG94 44427519 IC50 > 10000 nM T47107 CY87UN 44456923 Ki = 234 nM T47107 CW0T1S 44456924 Ki = 1510 nM T47107 CS2CV1 44456938 Ki = 61.3 nM T47107 C1S8MC 44575685 IC50 = 37000 nM T47107 CY3HW5 46224684 IC50 = 1100 nM T47107 CLS29B 46872626 IC50 > 10000 nM T47107 C2O8RZ 46886323 IC50 > 1000 nM T47107 CHSF07 49806372 IC50 > 1000 nM T47107 CD2K4R 50908681 Ki > 1000000 nM T47107 CM42BY 51000510 Ki > 1000000 nM T47107 CHP06V 52948258 Ki = 80 nM T47107 CZF5T9 53262772 IC50 = 61970 nM T47107 CD4H3S 53354074 Ki = 725 nM T47107 C8NA4L 53384644 IC50 > 30000 nM T47107 CCM71K 54669828 Ki = 660 nM T47107 COH41P 58325285 IC50 > 1000 nM T47107 C1MR8Q 60097495 IC50 > 10000 nM T47107 CNL04P 60155126 Ki = 12 nM T47107 C56PUM 60155209 Ki = 5.5 nM T47107 CV63UL 67240318 IC50 > 10000 nM T47107 CU60JG 71718528 IC50 > 50000 nM T47107 CV70GZ 71728100 Ki = 0.69 nM T47107 C7Q0AD 76286479 IC50 = 13000 nM T47107 CZF0N7 76287389 IC50 = 7800 nM T47107 C28STM 76287526 IC50 = 23000 nM T47107 CRJ45X 135589980 IC50 > 33000 nM T47107 C0J3BN 135678111 IC50 > 50000 nM T47107 C26ESH 136060555 IC50 = 4900 nM T47107 C6VB3O 145925651 IC50 >= 5000 nM T47107 C2MD1Q 155513187 IC50 > 10000 nM T47107 D00ERW 44444843 Ki > 8750 nM T47107 D02KPV 37783 Ki = 1.58 nM T47107 D02XHC 448912 IC50 > 100000 nM T47107 D04AXH 11574614 Ki = 5200 nM T47107 D06ZCX 10455969 IC50 = 2000 nM T47107 D07OAT 456214 IC50 > 10000 nM T47107 D08JPU 3501 IC50 = 2 nM T47107 D0CM6T 11314340 Ki = 1200 nM T47107 D0D6DH 10125830 IC50 > 50000 nM T47107 D0H7DQ 6419755 IC50 > 1000 nM T47107 D0K5ZY 105000 Ki = 19.4 nM T47107 D0Q3NG 11715520 Ki > 8800 nM T47107 D0S7IE 11658882 Ki > 8800 nM T47107 D0TO6S 2396 IC50 = 30 nM T89361 D04AIT 5280445 IC50 > 300000 nM T89361 D05SBO 46220502 IC50 = 1.9 nM T89361 D0K8KX 5280343 IC50 = 25000 nM T89361 D00UZR 5330286 IC50 = 15 nM T89361 D05ADP 160355 IC50 = 24500 nM T89361 D08MXP 44631912 IC50 = 6 nM T89361 D0DX4J 67409219 IC50 < 100 nM T89361 D0LF1U 5287969 IC50 = 80 nM T89361 D0P0KN 16739650 IC50 > 100 nM T89361 C4MNG8 445840 IC50 = 71 nM T89361 CB2H4D 16037675 IC50 = 7.8 nM T89361 C9TU1O 16046126 IC50 = 12 nM T89361 CZ48LS 24825971 IC50 = 5600 nM T89361 CY8L7E 24896769 IC50 > 10000 nM T89361 C3VRO9 44557921 IC50 > 10000 nM T89361 CKL1V8 49798556 IC50 > 20000 nM T89361 CCL3R5 49867929 IC50 = 47000 nM T89361 C6BPR2 58985201 IC50 > 50000 nM T89361 CBE67N 71731769 IC50 > 10000 nM T89361 CB64IQ 72194525 IC50 = 3.33 nM T89361 CYG95S 72707651 IC50 = 50 nM T89361 CNP0V5 72707724 IC50 = 43 nM T89361 CU4A5Q 72707728 IC50 = 42 nM T89361 CZAM98 72707790 IC50 = 33 nM T89361 CP13FK 72707853 IC50 = 29 nM T89361 C7VA5U 78161839 IC50 > 10000 nM T89361 C8W9KV 91844733 IC50 = 34000 nM T89361 C8UL7Y 122657565 IC50 = 0.9 nM T89361 CHT7A6 122657605 IC50 = 4 nM T89361 C6J5BQ 122657629 IC50 = 3.7 nM T89361 C0NPF8 122657632 IC50 = 244.1 nM T89361 C63VIC 122667249 IC50 = 2.3 nM T89361 CEG56K 122667252 IC50 = 2.9 nM T89361 C1SDO8 122667293 IC50 = 2.9 nM T89361 CLHF95 122667296 IC50 = 1.6 nM T89361 C5R4PU 122667312 IC50 = 23.6 nM T89361 CAQP38 122667319 IC50 = 2.7 nM T89361 CAJH71 122667328 IC50 = 5.8 nM T89361 CSY3M0 122667329 IC50 = 1.8 nM T89361 CJU5O4 122667350 IC50 = 1.6 nM T89361 C09GPH 122667359 IC50 = 2.2 nM T89361 CW95MK 122667361 IC50 = 1.6 nM T89361 CZT1C4 122667385 IC50 = 4.4 nM T89361 CR5MA6 122667387 IC50 = 4 nM T89361 CVB7D2 129102568 IC50 = 46 nM T89361 C9BOH1 129102571 IC50 = 36 nM T89361 C4T9DH 129102574 IC50 = 11.2 nM T89361 CJ25TP 129102576 IC50 = 271 nM T89361 C8U9SE 129102577 IC50 = 19 nM T89361 CBOS93 129102582 IC50 = 339 nM T89361 C32QTR 129102589 IC50 = 12.7 nM T89361 C1GJQ3 129102591 IC50 = 22 nM T89361 CZAB64 129102594 IC50 = 28 nM T89361 CXO0V7 129102595 IC50 = 178 nM T89361 C6Y7VA 129102598 IC50 = 275 nM T89361 C72GIC 129102599 IC50 = 392 nM T89361 C8EIU5 129102600 IC50 = 2.4 nM T89361 C06GCP 129102608 IC50 = 752 nM T89361 CL0VI3 129102610 IC50 = 247.8 nM T89361 C3AM4Y 129102611 IC50 = 17.4 nM T89361 CSTL63 129102640 IC50 = 45.6 nM T89361 C5M7PZ 129102643 IC50 = 15.8 nM T89361 C1H5GP 129102646 IC50 = 18.7 nM T89361 C2LWZ1 129318964 IC50 > 10000 nM T89361 CW41KL 134135943 IC50 = 18 nM T89361 CFM28H 134144635 IC50 = 34 nM T89361 C5PE1B 134153020 IC50 = 28 nM T89361 C48DGU 134156416 IC50 = 23 nM T89361 C3DNL6 137349544 IC50 = 32100 nM T89361 CU9O3A 137628639 IC50 = 45 nM T89361 C25ERN 137631967 IC50 > 1000 nM T89361 C06JRX 137637094 IC50 > 1000 nM T89361 C1DK0P 137651391 IC50 > 1000 nM T89361 CV5H3Z 137657932 IC50 > 1000 nM T89361 CB98HD 145950262 IC50 = 33.21 nM T89361 C7PU6X 145956666 IC50 = 19.24 nM T89361 CJ4FO8 145957807 IC50 = 84.31 nM T89361 CR2GW6 145994117 IC50 > 5000 nM T89361 D00ERW 44444843 Ki > 1549 nM T89361 D00RIX 5280443 IC50 = 1700 nM T89361 D01MNK 25125014 IC50 = 35500 nM T89361 D01UYI 5281607 IC50 = 6000 nM T89361 D09OAH 73292 IC50 = 3400 nM T89361 D0G3TK 5280863 IC50 = 22000 nM T89361 D0GN5Z 5281295 IC50 = 2440 nM T89361 D0MF5Y 5281614 IC50 = 850 nM T06020 C0MNQ1 44585675 IC50 = 33000 nM T06020 C5CFI1 44585676 IC50 = 64000 nM T06020 C28EYX 44585677 IC50 = 49000 nM T06020 C5PC2D 44585680 IC50 = 239000 nM T06020 CAI50S 44585682 IC50 = 110000 nM T06020 CJPF50 44585683 IC50 > 250000 nM T06020 CJE3C5 44585685 IC50 = 67000 nM T06020 C07PMC 44585688 IC50 = 87000 nM T06020 CZN50E 44585689 IC50 = 23000 nM T06020 CAR5O7 44585711 IC50 = 1700 nM T06020 C9UA8F 44585712 IC50 = 2000 nM T06020 CNT9A2 44585715 IC50 > 250000 nM T06020 CFL1E4 44585721 IC50 = 2100 nM T06020 CGBP74 44585722 IC50 = 1000 nM T06020 C5C0DF 44585796 IC50 = 16000 nM T06020 COM6C3 44585815 IC50 = 122000 nM T06020 CN2UJ7 44585816 IC50 > 125000 nM T06020 CCP0Q9 44585817 IC50 = 1600 nM T06020 C3BG0H 44585818 IC50 = 2400 nM T06020 CMT41Z 44585819 IC50 = 5700 nM T06020 CUZ70Y 44585820 IC50 = 6200 nM T06020 CT68MF 44585821 IC50 = 1200 nM T06020 C3W7PQ 44585822 IC50 = 1300 nM T06020 CX46PQ 44585823 IC50 = 45000 nM T06020 C5KO7W 44585824 IC50 = 12000 nM T06020 C9LTO7 44585825 IC50 = 40000 nM T06020 C6L3GE 44585826 IC50 = 5500 nM T06020 C69ILF 44585828 IC50 = 4600 nM T06020 C7P3QW 44585829 IC50 = 150000 nM T06020 CO1EN9 44585830 IC50 = 6300 nM T06020 CFOZ86 44585831 IC50 = 85000 nM T06020 CT9WS8 44585832 IC50 = 27000 nM T06020 C4DJ9F 44585833 IC50 > 100000 nM T06020 C2JPY0 44585834 IC50 > 125000 nM T06020 CTK31F 44585835 IC50 = 57000 nM T06020 CC7S6B 44585836 IC50 > 125000 nM T06020 C7NS2P 44585837 IC50 = 14000 nM T06020 CT24VQ 44585838 IC50 = 2300 nM T06020 C1FZS8 44585839 IC50 = 660 nM T06020 C68LSG 44585840 IC50 = 7200 nM T06020 C3ZJ1W 44585841 IC50 = 640 nM T06020 C2NSC8 44585842 IC50 = 13000 nM T06020 CCO8T4 44585844 IC50 = 2200 nM T06020 CQD68H 44585845 IC50 = 530 nM T06020 CP68RD 44585846 IC50 = 620 nM T06020 CD3LM0 44585864 IC50 = 37000 nM T06020 C18QEX 44585865 IC50 = 38000 nM T06020 CGHJ67 44585866 IC50 = 23000 nM T06020 C50MFB 44585867 IC50 = 8000 nM T06020 CB1M5K 44585868 IC50 = 19000 nM T06020 CKA7Q8 46883958 IC50 = 1000 nM T06020 CBSA67 46883960 IC50 = 1900 nM T06020 CE3N9K 46883970 IC50 = 2.6 nM T06020 C2V5BH 46883973 IC50 = 4.8 nM T06020 CS03XN 73345660 IC50 = 16000 nM T06020 D0QR7C 25090771 IC50 = 570 nM T93344 D01AYJ 1549008 Ki = 30 nM T93344 D02RQU 54687 IC50 > 10000 nM T93344 D0L5WM 2157 IC50 = 12000 nM T93344 D0I3XW 6443223 IC50 = 20 nM T93344 CNS46Y 5362831 IC50 > 400000 nM T93344 CB26DK 5368962 IC50 = 100000 nM T93344 C8AYV7 9803536 IC50 = 30 nM T93344 C0T3PG 9866789 IC50 = 150 nM T93344 C5BRJ8 10003000 IC50 = 120 nM T93344 C7ZSD2 10027508 IC50 = 1000 nM T93344 CLTI92 10049923 IC50 = 520 nM T93344 CSV71H 10051039 IC50 = 270 nM T93344 CD2YX3 10094306 IC50 = 90 nM T93344 C1DAI5 10097424 IC50 = 210 nM T93344 CRB8S7 10320681 IC50 = 30 nM T93344 CJ4TC2 10320682 IC50 = 3000 nM T93344 CA1YF9 10321591 IC50 = 8000 nM T93344 CNAO57 10342792 IC50 = 100 nM T93344 CKHE96 10343384 IC50 = 1000 nM T93344 CPV63M 10343599 IC50 = 70 nM T93344 CXD1Y3 10343600 IC50 = 100 nM T93344 CRS38B 10344325 IC50 = 5000 nM T93344 CR8Q3L 10345926 IC50 = 10000 nM T93344 C75VQR 10365704 IC50 = 8000 nM T93344 CM6RT8 10387722 IC50 = 20000 nM T93344 CXW60Y 10410842 IC50 = 60 nM T93344 CQJ19M 10411264 IC50 = 70 nM T93344 CA27XQ 10411438 IC50 = 150 nM T93344 C71XDK 10413184 IC50 = 70 nM T93344 C3YL1M 10456289 IC50 > 10000 nM T93344 CIT78L 10457630 IC50 = 50 nM T93344 C18TMR 10478007 IC50 = 130 nM T93344 CBO17J 10481638 IC50 = 5000 nM T93344 C9VZ2W 11212382 IC50 > 400000 nM T93344 CL29DR 11744451 IC50 = 870 nM T93344 CX7C5N 11744673 IC50 = 400 nM T93344 CR54EQ 14544607 IC50 > 400000 nM T93344 C28QMW 14544610 IC50 > 400000 nM T93344 CURA43 14544611 IC50 = 400000 nM T93344 CL0SF2 14544612 IC50 > 400000 nM T93344 C2H4CI 14544614 IC50 = 60000 nM T93344 CCP1F2 14544616 IC50 > 400000 nM T93344 C4C9GE 14544622 IC50 > 400000 nM T93344 CL6TQ9 14701004 IC50 > 400000 nM T93344 CBO8D6 14701006 IC50 = 40000 nM T93344 C54FWE 14701008 IC50 = 4000 nM T93344 C8S6IW 15666831 Ki = 4000 nM T93344 CS98RO 15838669 IC50 = 255 nM T93344 C67UXR 15838670 IC50 = 330 nM T93344 C5J8KR 15838671 IC50 = 200 nM T93344 CAMF70 15838673 IC50 = 250 nM T93344 C03VOB 15838674 IC50 = 390 nM T93344 C1Z0LR 44265964 IC50 = 13000 nM T93344 C0KZ2V 44270471 IC50 = 100 nM T93344 CM27WG 44270510 IC50 > 100000 nM T93344 CS60QJ 44270529 IC50 = 960 nM T93344 CY48HC 44275418 IC50 > 400000 nM T93344 CMD31V 44275664 IC50 = 270000 nM T93344 CNH8D9 44276379 IC50 = 290 nM T93344 CID6K5 44276456 IC50 = 450 nM T93344 CJ0PO4 44276457 IC50 = 210 nM T93344 C5XN3I 44276458 IC50 = 90 nM T93344 C6HE7D 44276512 IC50 = 230 nM T93344 CTV28E 44276537 IC50 = 150 nM T93344 C0U5OH 44276539 IC50 = 170 nM T93344 CUW15T 44276544 IC50 = 170 nM T93344 C8HC9D 44276545 IC50 = 90 nM T93344 C4O9BF 44276560 IC50 = 300 nM T93344 C9W5JU 44276564 IC50 = 10000 nM T93344 C3UVO4 44276589 IC50 = 1800 nM T93344 CY92XG 44276608 IC50 = 200 nM T93344 CW9QB1 44276609 IC50 = 6400 nM T93344 C6Z0ND 44309360 IC50 = 500000 nM T93344 CFCP61 44309362 IC50 = 500000 nM T93344 C7H2IZ 44309381 IC50 = 500000 nM T93344 CLSN73 44309423 IC50 = 500000 nM T93344 CVAR97 44363366 IC50 = 32000 nM T93344 C0K5JM 44363369 Ki = 2400 nM T93344 D0V4FC 10411224 IC50 = 20 nM T93344 D0Z9PB 14379145 IC50 = 4000 nM T17143 D02UFQ 11620908 IC50 = 5700 nM T17143 D04AHQ 71721540 IC50 = 800 nM T17143 D0E3TC 44259 IC50 = 40.4 nM T17143 CEL61X 44229839 IC50 > 10000 nM T17143 C3VRO9 44557921 IC50 > 10000 nM T17143 CEBO91 71452977 IC50 > 10000 nM T17143 CZ31PU 71583657 IC50 = 870 nM T14834 D05DVP 5717 IC50 = 85000 nM T14834 D0E1WY 9853499 IC50 = 0.54 nM T14834 CXTE02 381598 IC50 = 48100 nM T14834 C8F1LG 5713130 IC50 = 1000 nM T14834 CSH5X8 9804496 IC50 = 40 nM T14834 CTZO12 9833099 IC50 = 1.8 nM T14834 CQ2BF7 9848070 IC50 = 800 nM T14834 CU5J1V 9874688 IC50 = 110 nM T14834 CX38IE 9934500 IC50 = 800 nM T14834 CG7IA0 9949350 IC50 > 10000 nM T14834 CXF43E 9956414 Ki = 15000 nM T14834 COW23P 9962675 IC50 = 1580 nM T14834 C8S0IG 10129207 IC50 = 650 nM T14834 CXEM82 10129469 IC50 = 26 nM T14834 CPG5J9 10129524 IC50 = 750 nM T14834 C03RTA 10129556 IC50 = 330 nM T14834 C20ANE 10153521 IC50 = 200 nM T14834 C30ULY 10153550 IC50 = 760 nM T14834 C86CJR 10153696 IC50 = 290 nM T14834 CM2AC3 10175654 IC50 = 510 nM T14834 C90HPI 10175665 IC50 = 390 nM T14834 CQ7XZ0 10175670 IC50 = 330 nM T14834 CAU20O 10175688 IC50 = 120 nM T14834 CNSG34 10175749 IC50 = 190 nM T14834 C5UR6P 10197184 IC50 = 300 nM T14834 C1X6QT 10218918 IC50 = 3000 nM T14834 CM5O6I 10218948 IC50 = 150 nM T14834 C06AWG 10218990 IC50 = 190 nM T14834 C2H8FG 10240432 IC50 = 600 nM T14834 CBZ6Q0 10290262 IC50 = 320 nM T14834 C9PRZ1 10290266 IC50 = 410 nM T14834 CLD9Y1 10290267 IC50 = 500 nM T14834 CQY52D 10290293 IC50 = 200 nM T14834 CZ92MJ 10290318 IC50 = 450 nM T14834 C9V4RT 10290348 IC50 = 100 nM T14834 C5L4YQ 10290439 IC50 = 200 nM T14834 C6ZYC8 10328085 IC50 = 3.1 nM T14834 CBV0Y9 10533215 IC50 = 72 nM T14834 C0G6LH 10533428 IC50 = 6.2 nM T14834 C41ICO 10556947 IC50 = 78 nM T14834 CFRW59 10557219 IC50 = 38 nM T14834 CLMX05 10557273 IC50 = 21 nM T14834 CJG42P 10580948 IC50 = 90 nM T14834 CQRN03 10605372 IC50 = 22 nM T14834 CL0M1W 10652466 IC50 = 165 nM T14834 CBXS53 10676984 IC50 = 2.1 nM T14834 CIA89F 10700085 IC50 = 69 nM T14834 C9Y6QJ 10700199 IC50 = 83 nM T14834 C53DOA 10747457 IC50 > 10000 nM T14834 C9Z3AQ 10795187 IC50 = 34 nM T14834 C0BWZ7 10819234 IC50 = 5.3 nM T14834 CZR73S 10842587 IC50 > 10000 nM T14834 CLZ7J3 11251471 IC50 = 110 nM T14834 C3B4WX 11271909 IC50 = 3000 nM T14834 CKQP62 11496930 IC50 = 120000 nM T14834 CVW43P 11497159 IC50 = 40000 nM T14834 CX3P8C 11497542 IC50 = 2000 nM T14834 CB0K9J 11497620 IC50 = 22000 nM T14834 CH7V9B 11502687 IC50 = 8000 nM T14834 CNT59G 11504684 IC50 = 11000 nM T14834 C4GTM0 11504869 IC50 = 800 nM T14834 CAVD52 11518850 IC50 = 2000 nM T14834 CNGV16 11519043 IC50 = 5000 nM T14834 C2R3UN 11524898 IC50 > 10000 nM T14834 CC0D9I 11532809 IC50 = 7.8 nM T14834 C74MEN 11540188 IC50 = 8000 nM T14834 C0LW5Z 11540746 IC50 = 2000 nM T14834 C1DMF0 11540936 IC50 = 26000 nM T14834 CEI1K5 11541275 IC50 = 20000 nM T14834 CP4V7M 11553564 IC50 > 10000 nM T14834 CIU21X 11554459 IC50 = 16 nM T14834 CAR0F1 11562559 IC50 = 2000 nM T14834 CNE3Q8 11569236 IC50 = 5000 nM T14834 CN2VJ8 11570339 IC50 = 18000 nM T14834 CG1J9Y 11570365 IC50 > 50000 nM T14834 COM24U 11577779 IC50 = 500 nM T14834 CLU2B0 11596966 IC50 > 10000 nM T14834 CV41YE 11599170 IC50 = 4000 nM T14834 CZ0R2V 11605391 IC50 = 1.1 nM T14834 CXFN57 11606342 IC50 = 2000 nM T14834 C6ZBO3 11612059 IC50 = 11 nM T14834 CD6FI3 11613547 IC50 = 38000 nM T14834 C2BQW6 11620682 IC50 = 1000 nM T14834 C8GTF1 11628032 IC50 = 20000 nM T14834 CSA4P7 11634910 IC50 = 2000 nM T14834 C2TZ7N 11635232 IC50 = 3000 nM T14834 CSXQ73 11635535 IC50 = 93000 nM T14834 CCS73H 11642326 IC50 = 30000 nM T14834 CX4J9L 11647468 IC50 = 1100 nM T14834 CI29GO 11656186 IC50 = 23000 nM T14834 C9XJ2Q 11657115 IC50 = 1000 nM T14834 C3IX4M 11668242 IC50 = 165000 nM T14834 C8I1VW 11670484 IC50 = 6000 nM T14834 CPQR28 11670893 IC50 = 0.9 nM T14834 CGU4C6 11676881 IC50 = 110 nM T14834 CA0M6E 11677500 IC50 = 40000 nM T14834 C3NRV4 11678127 IC50 = 1000 nM T14834 C7CK9P 11682816 IC50 > 10000 nM T14834 CQ4ZC0 11683813 IC50 = 380 nM T14834 C81EOV 11690296 IC50 = 120 nM T14834 CRY7X0 11690325 IC50 = 35 nM T14834 CEFV61 11691462 IC50 = 340 nM T14834 CTX83E 11699306 IC50 = 2000 nM T14834 CVB21N 11699550 IC50 = 6000 nM T14834 C9E5CZ 11705385 IC50 = 560 nM T14834 CRCF90 11706164 IC50 > 10000 nM T14834 C5Y9CW 11706415 IC50 = 7000 nM T14834 C5UCW6 11706512 IC50 = 33000 nM T14834 CYCP42 11713964 IC50 = 3000 nM T14834 CT64DA 11718385 IC50 = 4300 nM T14834 CM0S6X 11720602 IC50 = 3000 nM T14834 CIY5C3 11803244 IC50 = 49 nM T14834 CBYH95 12113700 IC50 = 160 nM T14834 C10XVG 12113710 IC50 = 170 nM T14834 C29XMR 12113712 IC50 = 360 nM T14834 CWL1Q4 12113885 IC50 = 100 nM T14834 CMK5N9 12113887 IC50 = 52 nM T14834 CC4UM1 12992902 IC50 = 5000 nM T14834 CD6XP8 15949063 IC50 = 200 nM T14834 C6Q0SF 15949064 IC50 = 10 nM T14834 CU2R7L 15949065 IC50 = 30 nM T14834 C2KSW0 15949066 IC50 = 22 nM T14834 CSX78J 15949164 IC50 = 13 nM T14834 C8NY0F 15949165 IC50 = 6 nM T14834 C2KD5C 15949166 IC50 = 20 nM T14834 CKY56Q 16114651 IC50 = 260 nM T14834 C05DSL 16114652 IC50 = 3000 nM T14834 CF1LX4 16114653 IC50 = 30000 nM T14834 CCZ42P 16114658 IC50 = 5000 nM T14834 C8O6DM 16114784 IC50 = 5000 nM T14834 CZR2L8 16114785 IC50 = 500 nM T14834 CP46GB 16114907 IC50 = 16500 nM T14834 CG8H6K 16115150 IC50 = 28000 nM T14834 CJ1Q9G 16115396 IC50 = 90000 nM T14834 CCJ1E6 16115397 IC50 = 18000 nM T14834 CU5S1Q 16115522 IC50 = 110 nM T14834 C73FKI 16115658 IC50 = 7000 nM T14834 C6U7RH 16115659 IC50 = 1200 nM T14834 CK87BY 16115936 IC50 = 2300 nM T14834 C76BYC 16116076 IC50 = 4200 nM T14834 CK6J4C 16116079 IC50 = 6700 nM T14834 C29MEJ 16116209 IC50 = 5500 nM T14834 CVP1A7 16116329 IC50 = 1600 nM T14834 C2HI0O 16116330 IC50 = 5900 nM T14834 C62EUD 16116331 IC50 = 4000 nM T14834 C4W8NX 16116333 IC50 = 120 nM T14834 CZYV83 16116460 IC50 = 2500 nM T14834 CS36FU 16116594 IC50 = 11000 nM T14834 CFLK16 18373290 IC50 = 2000 nM T14834 C1NV6E 18373296 IC50 = 20000 nM T14834 C0HRV3 18373300 IC50 = 400 nM T14834 C1N5UG 18373303 IC50 = 20000 nM T14834 C9FJ2E 18373313 IC50 = 15000 nM T14834 C40ZME 18373324 IC50 = 5000 nM T14834 C9TRN8 18373347 IC50 = 6000 nM T14834 C5GXB8 18373357 IC50 = 900 nM T14834 CYP40J 18373370 IC50 = 38000 nM T14834 C94EQS 18373374 IC50 = 1000 nM T14834 CJZB94 18373404 IC50 = 17000 nM T14834 CDM6Q7 18373405 IC50 = 600 nM T14834 C9U1AF 21962244 IC50 = 200 nM T14834 C1WE4X 21962249 IC50 = 700 nM T14834 CD9PM8 21962250 IC50 = 300 nM T14834 CZ1QO3 21962257 IC50 = 490 nM T14834 CB01SD 21962284 IC50 = 600 nM T14834 CWH8K3 21962302 IC50 = 270 nM T14834 C54XJW 21962303 IC50 = 350 nM T14834 CRH74A 21962316 IC50 = 350 nM T14834 CRH8B4 21962325 IC50 = 150 nM T14834 CM3Z7W 21962341 IC50 = 350 nM T14834 CI1TK3 21962374 IC50 = 550 nM T14834 CKDS90 21962391 IC50 = 140 nM T14834 C50OHV 21962396 IC50 = 250 nM T14834 C93HRT 21962404 IC50 = 180 nM T14834 CY03BO 21962414 IC50 = 270 nM T14834 CWKY41 21962423 IC50 = 600 nM T14834 CVOE26 21962435 IC50 = 120 nM T14834 C5EIW2 21962461 IC50 = 170 nM T14834 C5UBG2 21962476 IC50 = 220 nM T14834 C4KP1Z 21962481 IC50 = 220 nM T14834 C9C3QJ 21962483 IC50 = 240 nM T14834 C1KU7G 21962516 IC50 = 470 nM T14834 C6NX0L 21962528 IC50 = 380 nM T14834 C78XUT 21962561 IC50 = 130 nM T14834 CK2E8O 24852608 IC50 = 330 nM T14834 C95YRL 24970330 IC50 = 28 nM T14834 CI61BV 25052581 IC50 = 75 nM T14834 C28IWR 25052583 IC50 = 11 nM T14834 CQ2T7N 25052600 IC50 = 140 nM T14834 C4L8JU 25052602 IC50 = 14 nM T14834 C3Z4VB 25052603 IC50 = 20 nM T14834 CVD8K0 25113744 IC50 = 300 nM T14834 CIO1A2 25222894 IC50 = 450 nM T14834 CMOF58 25223398 IC50 = 150 nM T14834 CQ5RF2 25224203 IC50 = 250 nM T14834 CNBT53 25230917 IC50 = 210 nM T14834 CO9H7F 25230919 IC50 = 22 nM T14834 C96BMU 44138105 IC50 = 5 nM T14834 CZVN40 44265843 IC50 = 420 nM T14834 CHPU37 44323712 IC50 = 40000 nM T14834 CGJ0R2 44359392 IC50 = 4500 nM T14834 CFR98A 44359397 IC50 = 2100 nM T14834 CFLG07 44359399 IC50 = 3600 nM T14834 CPK0R9 44359411 IC50 = 1900 nM T14834 C81SUL 44359643 IC50 = 24000 nM T14834 CY32KH 44359649 IC50 = 41000 nM T14834 CLIK19 44359651 IC50 = 400 nM T14834 C6TDF2 44378991 IC50 = 17000 nM T14834 CNE91J 44379002 IC50 = 2000 nM T14834 CL63QP 44379005 IC50 = 4000 nM T14834 C9TQ4K 44379017 IC50 = 14000 nM T14834 CYZL41 44379020 IC50 = 17000 nM T14834 CVA6Q4 44379093 IC50 = 8000 nM T14834 CVXJ07 44379109 IC50 = 7000 nM T14834 C5ZBU2 44406733 IC50 = 85000 nM T14834 CH57IW 44406736 IC50 = 90000 nM T14834 CN49PT 44406738 IC50 = 120000 nM T14834 CU84XN 44406746 IC50 = 340000 nM T14834 CH7F6Q 44410407 IC50 = 38700 nM T14834 C6BE4J 44411695 IC50 = 6700 nM T14834 C0KCR8 44411711 IC50 = 2400 nM T14834 CZB0H8 44411722 IC50 > 50000 nM T14834 CAU4S7 44411723 IC50 > 50000 nM T14834 CN9F8Z 44411726 IC50 = 27000 nM T14834 C95SVJ 44411730 IC50 > 50000 nM T14834 CN5YM2 44411736 IC50 = 30000 nM T14834 CA3P4Z 44411749 IC50 = 12400 nM T14834 CV28SP 44411754 IC50 > 50000 nM T14834 C9OG6Q 44411758 IC50 = 1600 nM T14834 C9VU2N 44411759 IC50 = 1300 nM T14834 CZ58SX 44411915 IC50 > 50000 nM T14834 COZ8S7 44411916 IC50 = 23000 nM T14834 C9DE2P 44411938 IC50 = 5000 nM T14834 CN4IG5 44411940 IC50 = 5600 nM T14834 C2PZD4 44411964 IC50 = 3500 nM T14834 CKN6B1 44411980 IC50 = 1300 nM T14834 C90PDS 44411986 IC50 > 50000 nM T14834 C8K6SL 44411989 IC50 = 7500 nM T14834 C1OIU8 44428715 IC50 = 370 nM T14834 COZU04 44428716 IC50 = 840 nM T14834 C4PFU1 44428717 IC50 = 500 nM T14834 CBQM79 44428718 IC50 = 390 nM T14834 CY0GE1 44428719 IC50 = 310 nM T14834 CD6IK1 44428720 IC50 = 500 nM T14834 CB68RV 44428725 IC50 = 1100 nM T14834 C5QO9W 44452129 IC50 = 2100 nM T14834 CA6G1W 44452131 IC50 = 600 nM T14834 CB0G1U 44452156 IC50 = 3300 nM T14834 CUM23Q 44452235 IC50 > 10000 nM T14834 CO8V5Z 44452260 IC50 = 500 nM T14834 CGQ8I0 44452261 IC50 = 1500 nM T14834 CXT53K 44452290 IC50 = 400 nM T14834 C7C6SQ 44452316 IC50 = 10000 nM T14834 CG8KR2 44452345 IC50 > 10000 nM T14834 C2Z4XT 44456454 IC50 = 100 nM T14834 CRA3J1 44564173 IC50 = 250 nM T14834 CH8R3J 44564174 IC50 = 350 nM T14834 CT9S1W 44591618 IC50 = 150 nM T14834 C3JC2D 44591640 IC50 = 85 nM T14834 C0F3TO 44591641 IC50 = 26 nM T14834 CLU6Z7 44591642 IC50 = 16 nM T14834 C5F8MI 44591673 IC50 = 26 nM T14834 C2AKU5 45102612 IC50 = 12 nM T14834 C6AJS1 46230394 IC50 = 8200 nM T14834 CW9HU1 46230442 IC50 = 1800 nM T14834 CI13KC 46230443 IC50 > 10000 nM T14834 C80OIN 46230444 IC50 = 5300 nM T14834 CNF42I 46230445 IC50 > 10000 nM T14834 C2BM0Y 46230536 IC50 > 10000 nM T14834 CQN6L9 46230537 IC50 = 2200 nM T14834 CUHD15 49851171 IC50 = 10 nM T14834 CIF3R0 49851262 IC50 = 71 nM T14834 CMDV01 49851263 IC50 = 10 nM T14834 CD5UA6 59317742 IC50 = 15 nM T14834 C4Z0HU 59317743 IC50 = 16000 nM T14834 C2NKI5 59317761 IC50 = 1000 nM T14834 CF9S8I 59317762 IC50 = 13000 nM T14834 CVD23X 59317780 IC50 = 720 nM T14834 C8RJ3X 59317788 IC50 > 100000 nM T14834 CG4BP6 59317805 IC50 = 1200 nM T14834 CD6MH5 59317813 IC50 = 130 nM T14834 CZNJ51 59317830 IC50 = 77 nM T14834 CTXH43 59317841 IC50 = 7 nM T14834 CR20ZD 59317843 IC50 = 570 nM T14834 CY06DJ 59317848 IC50 = 320 nM T14834 CYI9H0 59317854 IC50 = 180 nM T14834 CXO1C5 59317869 IC50 = 780 nM T14834 CWB05G 59317871 IC50 = 190 nM T14834 CC2WK7 59317878 IC50 = 980 nM T14834 C9NY3Q 59317892 IC50 = 26 nM T14834 C92ZOW 59317900 IC50 = 1400 nM T14834 C5XR9E 59317914 IC50 = 1200 nM T14834 C0LE7H 59317915 IC50 = 58 nM T14834 C1SX5U 59317921 IC50 = 36 nM T14834 C9J5GI 59317927 IC50 = 7 nM T14834 C37RAE 68517943 IC50 = 10000 nM T14834 C1P5FA 73387420 IC50 = 15 nM T14834 CBY93E 73387421 IC50 = 23 nM T14834 CND8T3 77847624 IC50 = 1200 nM T14834 C3RNM0 118711986 IC50 = 3900 nM T14834 CK4RO0 118711988 IC50 = 15000 nM T14834 C0K3GB 118711989 IC50 = 1700 nM T14834 C3DKC0 118711991 IC50 = 400 nM T14834 CK6CG0 118711992 IC50 = 1600 nM T14834 CK7J4X 118712624 IC50 = 300 nM T14834 C9WL2U 136118005 IC50 = 3500 nM T14834 CQTU94 137631367 IC50 = 31 nM T14834 CC4QL3 137660737 IC50 = 49 nM T14834 CMU3G9 154724033 IC50 = 22000 nM T14834 D02GTZ 44410505 IC50 = 8420 nM T14834 D03NYE 9906670 IC50 = 4400 nM T14834 D05LWK 44410408 IC50 = 11900 nM T14834 D07VJT 23661736 IC50 = 16800 nM T14834 D0F9PM 10290302 IC50 = 10 nM T14834 D0H6FG 10429254 IC50 = 640 nM T14834 D0J8TY 5280436 IC50 = 2300 nM T14834 D0L6GV 11962186 IC50 = 6000 nM T14834 D0P5UW 204106 IC50 = 150 nM T14834 D0W4VM 9846199 IC50 = 11 nM T14834 D0Y2BD 46230393 IC50 = 500 nM T11309 D0B5LF 448042 IC50 = 2630.27 nM T11309 D03KKR 3547 IC50 = 6918.31 nM T11309 C6HD4P 11295434 Ki = 33 nM T11309 CKEM34 11397616 Ki = 437 nM T11309 CYK18E 44573412 Ki = 110 nM T11309 C3AG9N 44573485 Ki = 6.8 nM T11309 CR3XS9 44573487 Ki = 31 nM T11309 CP9HC7 44573568 Ki = 50 nM T11309 CRY96M 53321650 IC50 > 31622.78 nM T11309 CPN53D 72702874 Ki = 6.1 nM T11309 C86HIK 72702875 Ki = 29 nM T11309 CRH15J 72702877 Ki = 18 nM T11309 CLJ1O9 72702878 Ki = 3.6 nM T11309 C4DIV8 72703068 Ki = 55 nM T11309 CON2L3 72703069 Ki = 54 nM T11309 C52QXT 72703070 Ki = 130 nM T11309 C4EQ1N 72703071 Ki = 3.9 nM T11309 CKMH39 72703272 Ki = 6.3 nM T11309 CJ6ZL0 72703273 Ki = 27 nM T11309 CC29GP 72703274 Ki = 35 nM T11309 C3MT0F 72703491 Ki = 2400 nM T11309 CEGB49 72703493 Ki = 134 nM T11309 CKD8G9 72705826 Ki = 43 nM T11309 CP76OK 72705827 Ki = 86 nM T11309 CPO89M 72705828 Ki = 70 nM T11309 D0L1UK 3064778 IC50 = 6918.31 nM T02551 D01AZG 5073 Ki = 6.7 nM T02551 D01FFA 72301 Ki = 1371 nM T02551 D01ZII 2726 Ki = 1.585 nM T02551 D03DJL 6918554 Ki = 1048 nM T02551 D03ELL 2159 Ki = 3.981 nM T02551 D03KQF 4011 Ki = 504 nM T02551 D03QGM 5355 Ki = 8 nM T02551 D04JCN 47811 Ki = 0.8511 nM T02551 D04KJO 3410 Ki = 1626 nM T02551 D05MBZ 129211 Ki = 0.28 nM T02551 D05XGO 11154555 Ki = 0.085 nM T02551 D05ZIK 4205 Ki > 20 nM T02551 D06YFA 31101 Ki = 87 nM T02551 D07MEH 3033769 Ki = 3.7 nM T02551 D08VYV 4168 Ki = 27 nM T02551 D0AJ5L 4615 Ki = 62.7 nM T02551 D0AV3G 3151 Ki = 3.5 nM T02551 D0B0CP 667467 Ki = 4.56 nM T02551 D0CQ0Z 33630 Ki = 136 nM T02551 D0D1AL 3559 IC50 = 0.06 nM T02551 D0G8NN 119570 Ki = 0.7244 nM T02551 D0H3HM 60795 Ki = 1 nM T02551 D0H6QU 6005 Ki = 2.6 nM T02551 D0H7KF 5002 Ki = 251.19 nM T02551 D0I8FI 3779 Ki = 4700 nM T02551 D0J5RN 9690109 Ki = 39000 nM T02551 D0KS6W 7077 Ki > 10000 nM T02551 D0L5YV 5152 Ki = 1049 nM T02551 D0P1FO 16078 EC50 = 10.2 nM T02551 D0P5SA 3372 Ki = 3.21 nM T02551 D0R1JV 60854 Ki = 6.31 nM T02551 D0R6RO 4184 Ki = 2841 nM T02551 D0R9EQ 5095 Ki = 2.9 nM T02551 D0T6QX 5736 Ki = 6.4 nM T02551 D0T7OW 681 EC50 = 0.11 nM T02551 D0U2OO 2477 Ki = 660 nM T02551 D0U5OE 3964 IC50 = 22 nM T02551 D0V4QS 135398745 Ki = 19.95 nM T02551 D0WV3U 4893 Ki > 7100 nM T02551 D0X7KB 28864 Ki = 0.1413 nM T02551 D0X7QQ 16363 Ki = 0.29 nM T02551 D0Y5UG 2160 Ki = 206 nM T02551 D0Y7XC 5374 Ki = 67.61 nM T02551 D0Z1RV 135398737 Ki = 88 nM T02551 D00POS 9931976 Ki > 50 nM T02551 D01GEB 219050 Ki = 0.4 nM T02551 D03RIO 24743758 Ki = 1.259 nM T02551 D07YVK 9818479 EC50 = 186 nM T02551 D0A7KI 3037308 Ki = 5.4 nM T02551 D0C8PE 16058752 Ki = 1159 nM T02551 D0L3JI 188942 Ki > 8000 nM T02551 D0LI1C 44469321 IC50 > 10000 nM T02551 D0N1HW 5311200 Ki = 380.19 nM T02551 D0W5EH 6918388 IC50 < 6 nM T02551 D0X2XF 177336 Ki < 1000 nM T02551 D00MQS 9926143 Ki = 424 nM T02551 D04UXX 3075615 Ki = 13.7 nM T02551 D07YLK 4350931 Ki = 25.9 nM T02551 D0K5EE 9868452 Ki = 0.3162 nM T02551 D0Q3GV 15389743 EC50 = 2.291 nM T02551 D01RAE 133079 Ki > 2778 nM T02551 D01WJZ 60820 Ki = 1.8 nM T02551 D01ZSF 24840389 Ki = 1.3 nM T02551 D02FNU 56971 IC50 = 1200 nM T02551 D02JMI 9888211 Ki = 0.7943 nM T02551 D03YPJ 5163 Ki < 10000 nM T02551 D03ZZH 9887537 Ki = 3.981 nM T02551 D06DZI 107780 Ki > 10000 nM T02551 D07ODD 132891 Ki = 985 nM T02551 D0A3OF 10026300 IC50 = 29 nM T02551 D0B7SP 11292933 Ki = 199.53 nM T02551 D0EE6L 3038495 Ki = 0.3 nM T02551 D0FH3X 9916104 Ki = 2.9 nM T02551 D0M7LV 5761 Ki = 27 nM T02551 D0M9GE 53389 Ki > 8000 nM T02551 D0OS6O 60149 Ki = 2.6 nM T02551 D0Q2JS 10436045 Ki = 7.943 nM T02551 D0TH1Z 57533 Ki = 0.16 nM T02551 D0UZ1I 9841864 Ki = 3.162 nM T02551 D0Y6SN 5311096 Ki = 3.981 nM T02551 D0YP7L 6604889 Ki = 2511.89 nM T02551 D0Z2WQ 57242 Ki = 0.9333 nM T02551 D0Z7AW 9820261 Ki > 2000 nM T02551 C7ALK2 1240 Ki = 3.37 nM T02551 COJD92 1687 Ki = 5380 nM T02551 CF08KR 4885 Ki = 10 nM T02551 CW56ZA 5290 Ki = 101 nM T02551 C54IUQ 5357 Ki = 6.31 nM T02551 C5H9CN 9287 Ki > 10000 nM T02551 CVW5J9 10220 Ki = 37 nM T02551 CKZX76 13122 Ki = 10000 nM T02551 C9E6DA 21171 Ki = 433 nM T02551 C87UJB 21454 Ki > 3700 nM T02551 CFGH18 27620 Ki = 72 nM T02551 C34MDW 30133 Ki = 58.88 nM T02551 C8Y6DE 37461 Ki = 0.43 nM T02551 CJS51G 52919 Ki = 3.5 nM T02551 CY2F8T 55445 Ki = 132 nM T02551 CGB1S7 57532 Ki = 1 nM T02551 COI7E6 59227 Ki = 3.99 nM T02551 CBJ5R0 65340 Ki = 12.59 nM T02551 C5Y8HP 68663 Ki = 11 nM T02551 CYH3T7 71101 Ki = 43.2 nM T02551 C6MRZ3 91588 Ki = 500 nM T02551 C3VK5J 99601 Ki = 10000 nM T02551 C9NJK8 114876 EC50 = 5.32 nM T02551 C2U4GI 117370 Ki = 465 nM T02551 CKP25M 121881 Ki < 1000 nM T02551 CKR4N3 122065 Ki = 73 nM T02551 C9IBE6 125156 Ki = 343 nM T02551 CG21YH 127262 Ki > 1000 nM T02551 C5SWN1 127698 Ki = 16.6 nM T02551 CD2C0M 128054 Ki = 1.82 nM T02551 C26CPK 130402 Ki = 230 nM T02551 CY8W6U 131213 Ki = 3.8 nM T02551 C9WG8X 131559 EC50 = 21.8 nM T02551 CC58NU 132955 EC50 = 0.81 nM T02551 C9YA8O 134002 Ki = 5.91 nM T02551 C6CW2T 151086 Ki = 831.76 nM T02551 C1ND9W 161665 Ki = 1713 nM T02551 C9OD2N 163091 Ki = 9.4 nM T02551 CLK7P3 169713 IC50 > 10000 nM T02551 CRL1X5 178078 Ki = 0.52 nM T02551 C2LS9I 182600 Ki = 83.5 nM T02551 CN85OB 224518 Ki = 10000 nM T02551 CFU89K 229971 Ki = 1419 nM T02551 C6B2XL 229972 Ki = 442 nM T02551 C5RC4G 231915 Ki = 42.7 nM T02551 C54MBU 304988 Ki = 10000 nM T02551 CO9CV0 305306 Ki = 10000 nM T02551 C7P5UY 319767 Ki = 1000 nM T02551 CKO65R 326582 Ki = 10000 nM T02551 CN1AP3 327142 Ki = 10000 nM T02551 CDP6K3 336212 Ki = 10000 nM T02551 C9XBO8 336213 Ki = 2412 nM T02551 CO70CY 338743 Ki = 10000 nM T02551 C06TFG 345239 Ki = 1381 nM T02551 CHZ1P6 380039 Ki = 60.1 nM T02551 CL4X9J 408500 Ki = 10000 nM T02551 CI5J0G 408574 Ki = 1258 nM T02551 CB9Q3U 409671 Ki = 10000 nM T02551 CF5CS4 410922 Ki = 2420 nM T02551 CC1BU0 422809 Ki = 297 nM T02551 CQOM79 424716 Ki = 429 nM T02551 C9F7CR 424721 Ki = 10000 nM T02551 CW5BE2 426310 Ki = 2615 nM T02551 CG2JX9 440229 Ki = 37.3 nM T02551 CV6D3N 443374 Ki = 5.012 nM T02551 C28ARG 511482 Ki = 150 nM T02551 CG59VA 511484 Ki > 400 nM T02551 C97TAX 516222 IC50 = 2700 nM T02551 C65AZI 516264 IC50 = 4000 nM T02551 CGIY90 688272 Ki = 88 nM T02551 CU8H9L 749986 Ki = 4400 nM T02551 CD7P8Y 763194 Ki = 1899 nM T02551 C6QLR0 763343 Ki = 1648 nM T02551 CLR75J 763625 Ki > 10000 nM T02551 C5SXQ1 763774 Ki > 10000 nM T02551 C9IK2J 792265 Ki = 59 nM T02551 C13TYL 792460 Ki = 112 nM T02551 C4AY9X 792584 Ki = 42 nM T02551 CW0CU9 798232 Ki > 10000 nM T02551 C08WCU 851833 Ki = 197.4 nM T02551 C9CZJ1 857428 Ki = 1600 nM T02551 CKG0A5 1158941 Ki = 1435.7 nM T02551 CJ30IQ 1248739 Ki = 3100 nM T02551 CM1TH8 1438298 Ki = 11000 nM T02551 C6N8EF 2812861 Ki = 1530 nM T02551 C3DN1I 2822063 Ki = 47.3 nM T02551 C64CZV 3038494 Ki = 0.9 nM T02551 C6Z4QI 3050372 Ki = 79.3 nM T02551 C5NA6S 3069135 Ki = 207 nM T02551 CBL51N 3156990 Ki = 2500 nM T02551 C82GMT 3246443 Ki = 82.4 nM T02551 C0U6EW 3504099 Ki = 103 nM T02551 C0YXV3 3676358 Ki > 10000 nM T02551 CD76NG 3691783 Ki = 193 nM T02551 CK3W2U 3716121 Ki = 83 nM T02551 C9J5YC 3746693 Ki = 820 nM T02551 CO0FZ1 4064342 Ki = 700 nM T02551 CY7PH0 4302960 Ki = 0.3162 nM T02551 CS6P5D 4797946 EC50 = 6354 nM T02551 CWB9I2 4987774 Ki = 31.8 nM T02551 C6FM8G 5029739 Ki = 480 nM T02551 C9AZ2I 5249956 Ki = 47.5 nM T02551 CMX45W 5311346 Ki = 1.4 nM T02551 C9FYP1 5312124 Ki = 1.259 nM T02551 C8RK1C 6086459 Ki = 1000 nM T02551 C8R4JX 6305587 Ki = 1.85 nM T02551 CXP45C 6430941 EC50 > 1000 nM T02551 C6L9DT 6466372 EC50 = 5581 nM T02551 CWNZ35 6469693 Ki = 3900 nM T02551 CJTQ40 6469918 Ki = 8800 nM T02551 CXZ53N 6603866 Ki = 179 nM T02551 CKP56W 6603867 Ki = 0.57 nM T02551 C54GCX 6604356 Ki = 3.467 nM T02551 C5WH0F 6604868 Ki > 2000 nM T02551 C0QCK1 6918455 Ki = 501.19 nM T02551 CW0ZE5 6918542 Ki = 80 nM T02551 CC5PQ0 6918601 Ki = 3700 nM T02551 C1WXY3 6918603 Ki < 1584.89 nM T02551 CD0Z4I 6918648 Ki = 199.53 nM T02551 C1R4IO 6937303 Ki = 2050 nM T02551 C6MR7E 8529065 Ki > 400 nM T02551 C3NK0H 8690650 Ki > 400 nM T02551 C07UXF 9268266 EC50 = 710 nM T02551 CVF3N1 9475051 EC50 = 114 nM T02551 C5FUS9 9795741 Ki = 1305 nM T02551 CCM0S1 9796255 Ki = 8.3 nM T02551 CUD06Z 9796627 Ki > 3500 nM T02551 CX3OB9 9797200 Ki = 2682 nM T02551 CXDA07 9797306 Ki > 8000 nM T02551 CY6WB3 9797495 Ki = 3900 nM T02551 CE0DI5 9804612 Ki = 3981.07 nM T02551 C8XGV3 9804849 IC50 = 2300 nM T02551 CNX4F0 9805456 Ki < 1995.26 nM T02551 C59RXH 9816005 Ki = 249 nM T02551 CV5L1J 9817253 Ki = 4.1 nM T02551 C6V0MU 9817774 Ki = 2 nM T02551 CWOS30 9817810 Ki = 940 nM T02551 C2V7HU 9819770 Ki = 2682 nM T02551 CQE93H 9820085 Ki > 3000 nM T02551 CR17LP 9820313 Ki = 263 nM T02551 CVMR82 9820327 Ki = 1 nM T02551 C1HNW6 9820680 Ki = 41.8 nM T02551 CL38GM 9826580 Ki = 0.4 nM T02551 C0AU9L 9826801 Ki = 1200 nM T02551 C8LP9E 9827991 Ki = 0.5 nM T02551 C8EC9B 9828617 Ki = 0.631 nM T02551 C2F5OX 9828632 Ki = 8 nM T02551 COG0R8 9836900 Ki = 10.4 nM T02551 C2MN0P 9837094 Ki = 2948 nM T02551 CWB61S 9838572 Ki = 224 nM T02551 CBN06W 9839050 Ki = 84 nM T02551 C4BPW7 9839426 Ki = 5 nM T02551 C8XER9 9840365 Ki = 220 nM T02551 C1U6ZX 9840672 Ki = 1.15 nM T02551 C7O0TI 9841203 Ki = 10 nM T02551 CF87HQ 9841608 Ki > 3000 nM T02551 C4B6JU 9847363 Ki = 0.02 nM T02551 C7S1YV 9849443 Ki = 10 nM T02551 C07TSW 9859120 Ki = 589.9 nM T02551 C7EZ2L 9859861 Ki > 10000 nM T02551 C4GT3Z 9861459 Ki = 0.4 nM T02551 CD12MS 9861786 Ki = 7.4 nM T02551 CNCK78 9862256 Ki = 300 nM T02551 C6ERH9 9863540 Ki > 3030 nM T02551 C0Q6AD 9863611 Ki = 15.85 nM T02551 CR06ME 9865584 Ki = 0.14 nM T02551 C5WYN4 9865858 Ki = 1.6 nM T02551 CB1F0C 9867475 Ki = 66 nM T02551 CJAU58 9868502 Ki = 1.259 nM T02551 CDFP50 9868793 IC50 = 489 nM T02551 C7AB8O 9870053 Ki < 10000 nM T02551 CQ4LC2 9872676 Ki = 1180 nM T02551 CL0F2R 9881980 Ki = 10 nM T02551 CY5HZ0 9882594 Ki = 260 nM T02551 COI69G 9883554 Ki > 3000 nM T02551 CW97YN 9883587 Ki = 60 nM T02551 C3DB5H 9884781 Ki = 2840 nM T02551 CTAC24 9885114 Ki = 679 nM T02551 CALV92 9886609 Ki = 29 nM T02551 CQ03IA 9887463 Ki = 0.4 nM T02551 CJW1P5 9888494 Ki = 1698.24 nM T02551 C9GB2M 9888555 Ki = 0.19 nM T02551 C6N8UE 9889681 Ki < 3162.28 nM T02551 CN6L8E 9889735 Ki = 6.31 nM T02551 C2XAH9 9889736 Ki = 10 nM T02551 CM52WU 9890119 Ki = 2511.89 nM T02551 CEG1K5 9891002 Ki < 1584.89 nM T02551 C7QMK5 9891617 Ki < 1000 nM T02551 CEL29O 9891618 Ki < 3981.07 nM T02551 C6WY0D 9891901 Ki = 0.233 nM T02551 C3J8GU 9892409 Ki = 1000 nM T02551 CAM25C 9894665 Ki = 62 nM T02551 CR8GO9 9902381 Ki = 2490 nM T02551 C1U3EY 9902382 Ki = 208 nM T02551 CUPI23 9903623 Ki = 95.5 nM T02551 C6RGI9 9904074 Ki = 1.4 nM T02551 CFI97S 9904205 IC50 = 169.82 nM T02551 CUN81Q 9905249 Ki = 3900 nM T02551 CYWQ50 9906447 Ki > 10000 nM T02551 CD3F4N 9906454 Ki > 3000 nM T02551 C7JFZ5 9906978 Ki = 200 nM T02551 CY51ZT 9907436 Ki = 0.22 nM T02551 C07SWP 9907461 Ki > 3000 nM T02551 C6YKE0 9908125 Ki = 870 nM T02551 C3NOI2 9909614 Ki = 1.5 nM T02551 CO7BK6 9909648 Ki = 240 nM T02551 C3BR6W 9910451 Ki = 1200 nM T02551 CXV7O3 9912796 Ki = 1.585 nM T02551 C78MDV 9913554 Ki = 316.23 nM T02551 C8LJ9H 9914930 Ki = 6.31 nM T02551 CE7UF1 9925530 Ki = 19.5 nM T02551 CJL38X 9925730 Ki = 94.6 nM T02551 C4UYZ7 9927441 Ki = 23 nM T02551 CP45YZ 9932385 Ki = 10 nM T02551 CUHL40 9933550 Ki = 19.95 nM T02551 CYVZ47 9934284 Ki = 501.19 nM T02551 CWO45F 9935387 Ki = 630.96 nM T02551 C1ES5F 9946469 Ki = 78.5 nM T02551 CZPM75 9948461 Ki = 17 nM T02551 CU2JM9 9948584 Ki = 1 nM T02551 C9EUM1 9948965 Ki = 347 nM T02551 CO2QA0 9949442 Ki = 450 nM T02551 CA07XW 9949531 Ki = 12.2 nM T02551 CIFG92 9949601 Ki > 3000 nM T02551 C02IMR 9949655 IC50 = 200 nM T02551 CXEZ63 9950165 Ki = 240 nM T02551 CZ6D4W 9951735 Ki = 140 nM T02551 CEL95F 9953774 Ki = 12.59 nM T02551 CK8NR2 9954121 Ki < 5011.87 nM T02551 CWSE34 9954899 IC50 = 53 nM T02551 CFR41N 9957068 Ki = 5.012 nM T02551 CZB52R 9967004 Ki = 839 nM T02551 CIW4R8 9968343 Ki = 864 nM T02551 CC1ZL3 9975465 Ki = 2270 nM T02551 CKU4N1 9976024 Ki = 49.7 nM T02551 CD8T5E 9976807 Ki = 220 nM T02551 CXT1W6 9977478 Ki = 0.42 nM T02551 CMYN90 9977532 Ki = 1.8 nM T02551 CL9F5W 9980760 Ki > 5000 nM T02551 CC6M7Z 9980998 Ki = 0.8 nM T02551 C4G1IX 9982854 Ki = 0.6918 nM T02551 CT7G0Y 9983212 Ki = 2.6 nM T02551 C56XEZ 9983667 Ki = 14.5 nM T02551 CB8NT0 9991216 Ki > 1362 nM T02551 C9BM2I 9991512 Ki = 83 nM T02551 CXQ5O2 9992189 Ki = 0.87 nM T02551 C8K6NO 9992903 Ki = 158 nM T02551 CB2EP7 9995264 Ki = 338 nM T02551 CUS7W9 9995379 Ki = 5.4 nM T02551 CP31VK 9995904 Ki = 1700 nM T02551 CV4BN3 9999267 Ki = 2.2 nM T02551 C6FA2J 10001207 Ki = 2100 nM T02551 C17ZTJ 10001256 Ki = 0.8 nM T02551 C50GJB 10003334 Ki > 4000 nM T02551 C1NQC9 10003809 Ki = 0.4571 nM T02551 CY53UZ 10003936 Ki = 0.45 nM T02551 CL9QS0 10004950 IC50 = 1930 nM T02551 C27WPA 10007017 Ki = 0.7413 nM T02551 C6TJI2 10009952 Ki = 28 nM T02551 CUX43N 10014136 Ki > 4762 nM T02551 CIX9P8 10014484 EC50 = 36 nM T02551 CUIQ94 10014924 EC50 = 1.1 nM T02551 C5ZJ4W 10015731 Ki = 2.87 nM T02551 CFP13M 10018300 Ki = 170 nM T02551 C9LC6Z 10020651 Ki > 2000 nM T02551 CXBN42 10021692 Ki = 1.6 nM T02551 C7MVE2 10027629 Ki = 11.8 nM T02551 CUC01W 10036468 EC50 > 5000 nM T02551 C9LF0P 10037311 Ki = 522 nM T02551 C3MK8V 10039198 Ki = 23 nM T02551 C1MJV4 10041417 Ki = 0.75 nM T02551 CN1M6G 10042972 Ki = 317 nM T02551 CUH63M 10046389 Ki = 2110 nM T02551 C8WPO6 10049549 Ki = 2691.53 nM T02551 CX27EK 10049758 IC50 = 8 nM T02551 CRZ48G 10050500 Ki = 3.162 nM T02551 CWGQ38 10052229 Ki = 79.43 nM T02551 CNU12A 10052433 Ki = 0.3162 nM T02551 C4GHO2 10053476 Ki = 0.55 nM T02551 CLNY93 10058787 Ki = 0.66 nM T02551 CFXB93 10059206 Ki = 1929 nM T02551 C5ZLK0 10060449 Ki = 86 nM T02551 CL23OT 10060538 Ki = 0.21 nM T02551 C6Y3NO 10063875 Ki = 2.4 nM T02551 C4PCO3 10065083 Ki = 244.1 nM T02551 CT2OG9 10065188 Ki = 177 nM T02551 CYX3E7 10065496 Ki = 8.72 nM T02551 C8Z6MA 10067306 IC50 > 5000 nM T02551 C4LQY1 10071413 Ki = 0.5754 nM T02551 C5HJ1G 10073022 Ki = 13.8 nM T02551 C03KWH 10073194 Ki = 2.6 nM T02551 C0V5ZR 10074155 Ki = 1.3 nM T02551 C75OQF 10075078 Ki = 2.512 nM T02551 CJ16VZ 10084583 Ki = 0.54 nM T02551 CX6L2Q 10086348 Ki = 2.6 nM T02551 C03CYX 10086395 Ki = 36 nM T02551 CGW9L7 10088259 Ki = 377 nM T02551 C2M6UR 10088426 Ki = 359 nM T02551 C0XB2Y 10090714 Ki = 31.4 nM T02551 CJXQ40 10092819 Ki = 0.92 nM T02551 CA3LE2 10098342 Ki = 3.467 nM T02551 CD3Y1G 10105186 Ki = 268 nM T02551 C7NK1P 10105359 Ki = 4.97 nM T02551 C54EYD 10108561 IC50 = 1659.59 nM T02551 CKCI50 10110263 Ki = 12 nM T02551 CVD86L 10130933 Ki = 28 nM T02551 C1DQ8L 10161526 Ki = 52 nM T02551 CV5FI6 10166896 Ki = 4 nM T02551 CP6Q1W 10173403 Ki = 15.85 nM T02551 CZ3RL4 10176243 Ki = 1520 nM T02551 C8M2KL 10178704 EC50 = 0.69 nM T02551 C2ZC0Q 10183626 Ki = 30 nM T02551 CZ97UO 10184153 Ki = 40 nM T02551 C7Y3JR 10200368 Ki = 14.2 nM T02551 CZKG96 10200496 Ki = 4.73 nM T02551 CFJY39 10216820 Ki = 6.31 nM T02551 CV1B7C 10217687 Ki = 0.7943 nM T02551 CWR4J6 10220541 Ki > 10000 nM T02551 CGJ5Q9 10225942 Ki = 15 nM T02551 C47KBM 10228202 Ki = 2.26 nM T02551 CS3X6I 10229397 Ki = 20 nM T02551 CO64WJ 10236758 Ki = 616.6 nM T02551 C8B4SV 10241065 Ki = 5890 nM T02551 COZ2S7 10242548 Ki = 136 nM T02551 C7LY2Z 10242819 Ki = 658 nM T02551 C5PDQ8 10242850 Ki = 339 nM T02551 CYCQ58 10245409 Ki = 250 nM T02551 CVF1E5 10246054 IC50 > 1000 nM T02551 CC3XF5 10247561 Ki = 8700 nM T02551 CFCP96 10247720 Ki = 7100 nM T02551 CY82IS 10248715 Ki > 4800 nM T02551 C6SB5G 10249134 Ki = 560 nM T02551 C4Q2SH 10249573 Ki = 1258.93 nM T02551 CC1PJ7 10251080 Ki = 3.9 nM T02551 C2UNO6 10251160 Ki = 19 nM T02551 CSPF93 10252272 Ki = 39.81 nM T02551 C6SNB5 10252580 Ki = 12.9 nM T02551 C7NO2S 10253333 Ki = 4.4 nM T02551 C9XTQ2 10253970 Ki = 4.5 nM T02551 COB28U 10254390 Ki = 0.13 nM T02551 CMRA02 10257042 Ki = 2511.89 nM T02551 C1FTS4 10263410 Ki = 1461 nM T02551 C5RF0W 10264090 Ki = 139 nM T02551 CE9Y8J 10276451 Ki = 0.5 nM T02551 C9MPY2 10300403 Ki = 19 nM T02551 C0L8VZ 10301202 Ki = 16 nM T02551 C8XKC0 10310103 Ki = 680 nM T02551 CJ3Q1T 10314824 Ki = 15000 nM T02551 C5R8TC 10315310 Ki = 30.9 nM T02551 C5XB6Y 10315866 Ki > 2000 nM T02551 CHYJ47 10317514 Ki = 18.9 nM T02551 CB8O9X 10318141 Ki = 966 nM T02551 CE6V0B 10330427 Ki = 1759 nM T02551 C57PKI 10330528 Ki = 777 nM T02551 C83GBY 10333405 Ki = 16.2 nM T02551 CRQN68 10333842 Ki = 1.2 nM T02551 C6WEU2 10334422 Ki = 59 nM T02551 CHJ4W9 10335148 Ki = 10 nM T02551 CNAV40 10340492 Ki = 44.7 nM T02551 C9IAV3 10346043 Ki > 5011.87 nM T02551 CBAZ60 10353207 Ki = 514 nM T02551 C0H3VS 10355305 Ki > 1285 nM T02551 CXO8I7 10355406 Ki = 4.42 nM T02551 CPK71L 10356389 Ki = 171 nM T02551 C1RX9F 10357631 Ki = 7 nM T02551 C1NTD8 10359539 Ki = 13000 nM T02551 CXAK13 10359942 Ki > 4400 nM T02551 C32KOP 10360923 Ki = 4400 nM T02551 CD4H6R 10361512 Ki = 21000 nM T02551 C2A5PV 10364677 Ki = 0.35 nM T02551 C0WVD9 10367857 Ki = 0.38 nM T02551 CJ6L9D 10368423 Ki = 3.9 nM T02551 CQEJ41 10368773 Ki = 3.981 nM T02551 C2X9PQ 10369220 Ki = 1.4 nM T02551 CH1IY6 10375676 Ki = 0.75 nM T02551 CD9OQ2 10377227 Ki = 2150 nM T02551 CIX51R 10378194 Ki = 850 nM T02551 CL48ZG 10380129 Ki = 1414 nM T02551 CR3KU9 10380133 IC50 > 5000 nM T02551 CDAC63 10381889 IC50 = 0.5495 nM T02551 C6DFI4 10382581 Ki = 2480 nM T02551 CEX1T3 10384736 Ki = 92 nM T02551 CER30L 10384998 Ki = 18.9 nM T02551 C7J2TY 10389636 Ki = 0.5012 nM T02551 CQ90WG 10390058 Ki = 3 nM T02551 CT3DJ5 10391240 Ki = 338 nM T02551 C4DZ0M 10392655 Ki = 2.1 nM T02551 C4UG3B 10395316 Ki = 5 nM T02551 CD5H6P 10397550 Ki = 631 nM T02551 C6J2ZL 10402378 Ki = 1601 nM T02551 CIF2V7 10402380 Ki = 23.8 nM T02551 C8WK6Q 10402381 Ki = 978 nM T02551 CJNR48 10403092 Ki = 1.98 nM T02551 CX2Y7J 10403608 Ki = 140 nM T02551 C4L5PQ 10404657 Ki = 491 nM T02551 C4OF7Y 10404663 Ki = 33 nM T02551 CS3OC4 10405678 Ki = 1136 nM T02551 CA2N8B 10406968 Ki = 149 nM T02551 CM50VF 10406989 Ki = 6.69 nM T02551 C04WGF 10407367 IC50 = 1558 nM T02551 CC5A2I 10411237 Ki = 0.18 nM T02551 CH5M7W 10413085 Ki = 0.2455 nM T02551 C4TPN1 10413595 Ki = 1000 nM T02551 CS6W9C 10414769 Ki = 1.259 nM T02551 C60ICT 10420915 Ki = 573 nM T02551 CCM6Y7 10421679 Ki = 40 nM T02551 C1EKY2 10422509 EC50 > 688 nM T02551 CZ5HC6 10425024 Ki = 24 nM T02551 CO76HW 10425969 Ki = 2350 nM T02551 CA3PI9 10427977 Ki = 4570.88 nM T02551 C4YBI9 10428654 Ki = 173 nM T02551 CL0ZB2 10430935 Ki = 65.9 nM T02551 C8ZA3G 10432808 Ki = 310 nM T02551 CD7U5I 10433930 Ki > 3981.07 nM T02551 C9A4MJ 10436285 Ki = 1.4 nM T02551 C4UN0A 10436653 Ki = 0.68 nM T02551 C8KD1B 10438027 Ki = 1.59 nM T02551 C8MF4H 10438351 Ki = 1.585 nM T02551 C9WB1M 10444260 EC50 > 10000 nM T02551 C1CO4G 10447709 Ki = 232 nM T02551 CL8HQ6 10450082 IC50 = 5600 nM T02551 CS1LF0 10450580 Ki = 3113 nM T02551 CVPK09 10450880 Ki = 2780 nM T02551 C1SZU3 10450892 Ki = 3.89 nM T02551 C9WS1O 10451844 Ki = 0.99 nM T02551 CW0ND4 10454026 Ki = 0.32 nM T02551 C04MGE 10454684 Ki = 6700 nM T02551 CUB9J6 10456040 Ki = 1.7 nM T02551 C05PSB 10456166 Ki = 0.6607 nM T02551 CK15JL 10456628 Ki = 1.9 nM T02551 CWE8U9 10457321 Ki = 24 nM T02551 CN6CD4 10457955 Ki = 10.4 nM T02551 CAM7K8 10458892 Ki = 627 nM T02551 CN41CS 10466682 EC50 = 32 nM T02551 C8RQZ4 10466922 Ki = 509 nM T02551 CZ8X1Q 10466923 Ki = 105 nM T02551 CM23NE 10467118 Ki > 1285 nM T02551 CV9N7G 10470579 Ki = 81 nM T02551 COV85C 10472143 Ki = 6 nM T02551 C5LBS7 10472158 IC50 > 5000 nM T02551 CUW3M2 10473658 Ki = 268 nM T02551 C05ZCT 10474964 Ki = 1570 nM T02551 CPI5M7 10476504 EC50 = 1.4 nM T02551 CE79QV 10477871 Ki = 0.2512 nM T02551 CEF2O6 10478367 Ki > 10000 nM T02551 CFLZ47 10479188 Ki = 65 nM T02551 CJI15O 10479214 Ki = 0.72 nM T02551 CCT42I 10479465 Ki = 1.13 nM T02551 CEP10Q 10479822 Ki = 0.3548 nM T02551 CD3A2O 10492351 Ki > 4400 nM T02551 C2WNH9 10494394 Ki = 190.55 nM T02551 C4JWB8 10494689 Ki = 19.7 nM T02551 CP51BI 10495881 Ki = 289 nM T02551 CG7Y1H 10497177 Ki = 550 nM T02551 C3ZW8P 10497179 Ki = 1100 nM T02551 C7VC6L 10497193 Ki = 920 nM T02551 CX1UD7 10498094 Ki = 1700 nM T02551 CHUF43 10498196 Ki = 428 nM T02551 CRUT74 10498972 Ki = 1698.24 nM T02551 C9M3FN 10499950 Ki = 54 nM T02551 CA1YR2 10502670 Ki = 0.251 nM T02551 CN9BT6 10512444 Ki = 0.71 nM T02551 C1NK6V 10515180 Ki = 1050 nM T02551 CN28AB 10515841 Ki = 3.58 nM T02551 C1GRL4 10518406 Ki = 369 nM T02551 CYL86S 10520941 Ki = 1200 nM T02551 C8ZMA1 10522334 Ki = 600 nM T02551 C12ZTU 10522613 Ki > 3200 nM T02551 C38ACZ 10522614 Ki = 130 nM T02551 CYP98E 10522950 Ki = 26 nM T02551 C7TZ3K 10524751 Ki = 1800 nM T02551 CI67OK 10535587 Ki = 2459 nM T02551 C59NSH 10543696 Ki > 8000 nM T02551 CU2E4W 10544865 Ki > 8000 nM T02551 C8ZG3C 10545941 Ki > 3030 nM T02551 CXI49Z 10546453 Ki = 2000 nM T02551 C7UCS1 10546540 Ki = 320 nM T02551 C40CJM 10546828 Ki = 1300 nM T02551 CYF64N 10547607 Ki > 3900 nM T02551 C4VZ2K 10549355 Ki = 1100 nM T02551 CQD6C8 10551026 Ki = 84 nM T02551 CBV9N4 10551197 Ki = 1.6 nM T02551 CH7E0W 10559624 Ki = 1.41 nM T02551 CKFH63 10560954 Ki = 158 nM T02551 CJH5T9 10567430 Ki = 3100 nM T02551 CC56ON 10568805 Ki = 591 nM T02551 CYL67U 10569690 Ki = 3600 nM T02551 C60SMR 10570080 Ki = 1100 nM T02551 C6S0TG 10570898 Ki > 3000 nM T02551 CTR45A 10570997 Ki = 590 nM T02551 C1YU3Q 10571927 Ki > 4000 nM T02551 CHE80N 10573876 Ki = 630.96 nM T02551 C02HSA 10574303 Ki = 15 nM T02551 C0O6IU 10586728 Ki = 199 nM T02551 C9SP3R 10587140 Ki = 3400 nM T02551 COL98E 10588194 Ki = 134.9 nM T02551 CP1Y7K 10589218 Ki = 66 nM T02551 C12ZRK 10590285 Ki = 234.42 nM T02551 CEH05N 10590717 Ki = 1400 nM T02551 CRJ13B 10593191 Ki = 174 nM T02551 C8E4HR 10593869 Ki = 1200 nM T02551 C97NMI 10594054 Ki = 920 nM T02551 CM7Z9X 10594113 Ki = 160 nM T02551 C17ZDI 10594242 Ki = 38 nM T02551 CD27FZ 10594764 Ki = 140 nM T02551 CDO93P 10595908 Ki = 46 nM T02551 C57DKO 10596380 IC50 = 350 nM T02551 CVZ10Y 10596978 Ki = 0.8 nM T02551 CO23YX 10597140 Ki = 1000 nM T02551 C6ECP0 10598935 Ki = 5 nM T02551 CU8DW9 10608413 Ki = 1450 nM T02551 C7GDX0 10612157 Ki = 1.1 nM T02551 CH49UB 10613605 Ki = 34 nM T02551 C3FS5U 10615437 Ki = 1400 nM T02551 C9JI3A 10615787 Ki = 95 nM T02551 C5XI7L 10616050 Ki = 2470 nM T02551 C56UGP 10617366 Ki = 830 nM T02551 CT5A6H 10617381 Ki = 49 nM T02551 CWQ76V 10617946 Ki = 240 nM T02551 C6QB8L 10618211 Ki = 510 nM T02551 C2LN0J 10618874 Ki > 4000 nM T02551 CJ7R5F 10618875 Ki = 430 nM T02551 CPJ0H3 10618928 Ki = 2300 nM T02551 C3VQK1 10619612 Ki = 360 nM T02551 CJ40ZT 10619737 Ki = 1200 nM T02551 CDZ16W 10620139 Ki > 3000 nM T02551 C1RXC5 10620194 Ki = 4.94 nM T02551 CKF8L2 10637198 Ki = 11 nM T02551 C0V5NM 10638052 Ki = 56 nM T02551 C8O4BC 10639430 Ki > 6665 nM T02551 C9D5MP 10640530 Ki = 491 nM T02551 CK4O3W 10641637 Ki = 6400 nM T02551 C2B5NL 10641783 Ki = 1790 nM T02551 C89NYU 10641954 Ki = 2620 nM T02551 C0DCY3 10641955 Ki = 2630 nM T02551 CKP3A1 10642106 Ki > 3030 nM T02551 CPTF56 10642239 Ki = 1450 nM T02551 CIFM84 10642428 Ki = 3.7 nM T02551 CED15G 10643588 Ki = 380 nM T02551 CL8KB3 10643589 Ki = 250 nM T02551 C4K0PA 10643780 Ki = 33000 nM T02551 CFC38D 10663221 Ki = 4400 nM T02551 CTP8L0 10664621 Ki = 232 nM T02551 C43FER 10665101 Ki = 464 nM T02551 CU3XJ4 10665598 Ki = 550 nM T02551 CI2OT7 10665626 Ki = 1300 nM T02551 C31ZOC 10666315 Ki = 220 nM T02551 CWE53T 10667201 Ki = 1900 nM T02551 C7K9DP 10667579 Ki > 4700 nM T02551 C4IY3Z 10667966 Ki = 2800 nM T02551 CQ2F1P 10679847 Ki = 35.8 nM T02551 CU31PH 10682854 Ki = 648 nM T02551 CO49AQ 10683127 Ki = 3003 nM T02551 CZLJ52 10684706 Ki = 234.42 nM T02551 C0ZCG1 10684789 Ki = 6.5 nM T02551 C6R7JD 10685891 Ki = 3.4 nM T02551 C7T2FU 10687362 Ki = 2210 nM T02551 CY4Z1R 10687967 Ki = 2100 nM T02551 CBW96O 10688035 Ki = 3600 nM T02551 C60DRH 10688036 Ki > 4200 nM T02551 CC1E7W 10690200 Ki = 930 nM T02551 CEM56L 10691523 Ki = 1300 nM T02551 CD1KF8 10691599 Ki = 80 nM T02551 CHZ8O2 10692886 Ki = 13.1 nM T02551 C8OC6U 10704110 Ki = 0.74 nM T02551 CU25LW 10708280 Ki = 169 nM T02551 C2OCP6 10711859 Ki > 8000 nM T02551 CE5QA3 10713620 Ki = 3.4 nM T02551 CG8KF5 10713960 Ki = 4.7 nM T02551 C4O6KG 10714184 Ki = 510 nM T02551 CHN8Q9 10725712 Ki = 150 nM T02551 CHN3T8 10729313 Ki = 8.62 nM T02551 C71VBX 10732925 Ki = 380.19 nM T02551 CO9BL7 10734727 Ki = 97.72 nM T02551 CHN4A3 10735344 Ki = 1200 nM T02551 CQ2DU0 10735405 Ki = 630 nM T02551 CO1DT0 10735463 Ki = 2980 nM T02551 C8VGB5 10736673 Ki = 89 nM T02551 CNWC38 10737474 Ki = 66 nM T02551 CY5HG9 10738530 Ki = 870 nM T02551 CSA67W 10738750 Ki = 48 nM T02551 C9RAU7 10739946 Ki > 4000 nM T02551 CI06WV 10740593 Ki = 0.02 nM T02551 C4I9VE 10756932 Ki = 800 nM T02551 C9Z8TB 10757990 Ki > 8000 nM T02551 C8XD2C 10758004 Ki = 177 nM T02551 C19UPY 10759511 Ki = 548 nM T02551 C21TFA 10759963 Ki = 56.7 nM T02551 CH5AY1 10760638 Ki = 600 nM T02551 CHN8T2 10760813 Ki = 720 nM T02551 CDNE69 10761258 Ki = 364 nM T02551 CC2L1A 10762432 Ki = 180 nM T02551 CAWG43 10765237 Ki = 32 nM T02551 C3LB9N 10780510 Ki = 72.44 nM T02551 CX4NK7 10780717 Ki = 0.36 nM T02551 CRUD74 10780928 Ki = 510 nM T02551 CU9T8V 10780942 Ki = 16.98 nM T02551 C4G8HB 10783874 Ki = 150 nM T02551 C1K4OD 10785202 Ki = 210 nM T02551 C6J2FC 10786367 Ki = 4300 nM T02551 C96NIC 10786891 Ki = 32 nM T02551 CXO6J4 10801405 Ki = 266 nM T02551 CL1CV6 10801925 Ki = 27.6 nM T02551 CP74YO 10803828 Ki = 0.2 nM T02551 CB74KW 10803829 Ki = 1 nM T02551 CB45KG 10805355 Ki = 345 nM T02551 C5M9AW 10806501 Ki > 4000 nM T02551 CS7YU8 10807795 Ki = 859 nM T02551 C24QAM 10809899 Ki = 220 nM T02551 CZ1F3B 10824155 Ki = 4400 nM T02551 C1SK9V 10826290 Ki > 1900 nM T02551 CJ9BY0 10827222 Ki = 20 nM T02551 CCN52S 10830557 Ki = 5200 nM T02551 C1QMR4 10831735 Ki = 13000 nM T02551 CJ1DI4 10831786 Ki = 1800 nM T02551 CM83SE 10833953 Ki = 20000 nM T02551 C8MHZ9 10835110 Ki = 1000 nM T02551 CF1S7E 10852461 Ki = 950 nM T02551 CPU26G 10854370 Ki > 3030 nM T02551 CI6PW4 10854386 Ki = 40 nM T02551 C9A8KN 10862425 Ki = 4.3 nM T02551 CHS8N5 10862670 Ki = 3.46 nM T02551 CL9Q3F 10863645 Ki = 37.2 nM T02551 CZYF05 10871118 Ki = 12000 nM T02551 CJ17GX 10874342 Ki = 2.96 nM T02551 CQ3TR7 10879566 Ki = 247 nM T02551 CMV36C 10884046 Ki = 18 nM T02551 CLEM91 10885047 Ki = 262 nM T02551 CD3U9P 10885524 Ki = 19 nM T02551 CRI50E 10885636 IC50 = 195 nM T02551 CV4ZO0 10894526 Ki = 0.5 nM T02551 CU80EA 10895106 Ki = 51 nM T02551 CMJD46 10895845 Ki = 1.28 nM T02551 CW8UH1 10905430 Ki = 0.64 nM T02551 C3X6QE 10906470 Ki = 10.2 nM T02551 CCHK19 10906679 Ki = 1.31 nM T02551 CX65PW 10907460 IC50 = 341 nM T02551 CL8AG5 10917920 Ki = 2900 nM T02551 C2UZ8H 10917953 Ki = 1400 nM T02551 CSM1Q2 10919602 Ki = 3.6 nM T02551 C6D7JR 10924369 Ki = 3570 nM T02551 CT79NZ 10927276 IC50 = 3180 nM T02551 C67FYJ 10927750 Ki = 1460 nM T02551 CN7C6W 10927912 Ki = 9.62 nM T02551 CH2OW6 10928654 Ki = 4.1 nM T02551 CU09AV 10937901 IC50 = 1910 nM T02551 C7AKH6 10939008 Ki = 1.8 nM T02551 CGZA42 10939167 Ki = 0.16 nM T02551 C0UGV5 10939222 Ki = 0.5012 nM T02551 C69ULE 10939408 Ki = 1.08 nM T02551 CPBA97 10939644 Ki = 0.43 nM T02551 C25TSY 10940279 Ki = 0.75 nM T02551 CC07JE 10942784 Ki = 5.12 nM T02551 CNB39C 10947658 Ki = 8 nM T02551 CN7XS4 10948527 IC50 = 160 nM T02551 C2SMP6 10949917 Ki = 0.56 nM T02551 CVN2Y8 10950916 Ki = 300 nM T02551 C1JD5K 10951105 Ki = 9.2 nM T02551 CJ5HP9 10951185 Ki = 19.5 nM T02551 C3JCI2 10960333 Ki = 12000 nM T02551 C2IGR9 10960767 Ki = 1.5 nM T02551 CBPS24 10961112 Ki = 1 nM T02551 CH14OY 10961938 Ki = 0.6 nM T02551 CUNX16 10971014 Ki = 0.6 nM T02551 C9DLO4 10971923 Ki = 7.99 nM T02551 C9HPJ3 10972865 Ki = 110 nM T02551 C5NRU3 10973768 Ki = 590 nM T02551 CE5PG3 10974122 Ki = 358 nM T02551 C6NF4A 10978080 Ki = 39.81 nM T02551 CFU1S9 10980338 Ki = 4900 nM T02551 C2HP7F 10981761 IC50 = 29 nM T02551 CJL0F7 10983103 Ki = 23.3 nM T02551 CB86ST 10983150 Ki = 7.8 nM T02551 CM9JY3 10988746 Ki = 60 nM T02551 C9AIQ2 10993488 Ki = 320 nM T02551 CNU2H3 10994539 Ki = 19.5 nM T02551 CS72LE 10994916 Ki = 1.2 nM T02551 CY3KA2 11005177 Ki = 42 nM T02551 CJC9K4 11005810 IC50 = 538 nM T02551 CO36VS 11005852 Ki = 28 nM T02551 CN32LJ 11015257 Ki = 108 nM T02551 C3FWN7 11016080 Ki = 100 nM T02551 C6BZR9 11016169 Ki = 2.5 nM T02551 CXZ29Y 11016342 Ki = 1.98 nM T02551 CH9GU5 11016418 Ki = 3100 nM T02551 CT56RB 11026289 Ki = 430 nM T02551 CGHN43 11027407 Ki = 7.8 nM T02551 C4Y9XK 11033734 Ki = 100 nM T02551 C01NDT 11036640 Ki = 645.65 nM T02551 CU6HR7 11036641 Ki = 16 nM T02551 C7C2RI 11044146 Ki = 108 nM T02551 C7KDU9 11048013 Ki = 140 nM T02551 CQ97YN 11048095 Ki = 0.73 nM T02551 C0N9VE 11048899 Ki = 40 nM T02551 C9FPV0 11048937 Ki = 6.3 nM T02551 CC1YO2 11049209 Ki = 2100 nM T02551 C0SUF4 11057969 Ki = 360 nM T02551 CTL9P3 11058442 Ki = 0.59 nM T02551 CE3J0B 11068912 Ki = 250 nM T02551 CP21DQ 11069795 Ki = 0.46 nM T02551 CG41BK 11071079 IC50 = 456 nM T02551 CUJ4W7 11071135 Ki > 7100 nM T02551 CVCE26 11076818 Ki = 117 nM T02551 CG63OS 11077918 Ki = 10000 nM T02551 CNF43K 11078813 Ki = 23000 nM T02551 CQ6W8Y 11091160 Ki = 0.38 nM T02551 CM2BD4 11092112 Ki = 2800 nM T02551 CN43SG 11102013 Ki = 0.44 nM T02551 C6TAH5 11102080 Ki = 32 nM T02551 CBM1I9 11102188 Ki = 0.55 nM T02551 C94EVP 11102206 Ki = 0.74 nM T02551 CW83IO 11102301 Ki = 0.68 nM T02551 CO5Y6W 11113582 Ki = 396 nM T02551 C7DE0U 11113605 IC50 = 977 nM T02551 CVE8T3 11121216 Ki = 150 nM T02551 CUN87A 11122812 Ki = 0.52 nM T02551 CTXS48 11133385 Ki = 340 nM T02551 CXP12A 11133602 Ki = 64 nM T02551 CUD5A0 11134444 Ki = 107 nM T02551 C0C3FI 11134596 Ki = 213 nM T02551 CU6PV0 11143820 IC50 = 2120 nM T02551 CQC54U 11145409 Ki = 700 nM T02551 CK7H9L 11146824 Ki = 92 nM T02551 C7EJX5 11150632 Ki = 60.26 nM T02551 CW7Y9O 11163741 Ki = 10 nM T02551 C56VFO 11166027 Ki = 2.2 nM T02551 C39PED 11177610 Ki = 0.8 nM T02551 C6CL1Y 11178830 Ki = 794.33 nM T02551 COI4G0 11186086 Ki = 24.2 nM T02551 C0W4SM 11186523 Ki = 15 nM T02551 CN06GJ 11186895 Ki = 262 nM T02551 C1QL8N 11197872 Ki = 2511.89 nM T02551 C9N5QU 11200511 Ki > 1000 nM T02551 CP8ZQ6 11203357 Ki = 3.2 nM T02551 CPX23W 11209208 IC50 > 10000 nM T02551 CXO67U 11213037 Ki = 0.28 nM T02551 CQ1E8L 11213136 Ki = 0.3162 nM T02551 C6D1MZ 11223004 Ki > 5000 nM T02551 CF08TL 11223885 Ki = 0.4 nM T02551 CN7CG0 11224283 Ki = 1.2 nM T02551 C1VM2S 11225043 Ki = 1 nM T02551 C6LB4S 11230330 EC50 = 2.4 nM T02551 CZ07AU 11231779 Ki = 7943.28 nM T02551 CZJ6O3 11243315 Ki = 323.59 nM T02551 CCKI68 11247894 Ki = 2.3 nM T02551 C90WSG 11248705 Ki = 1000 nM T02551 CHQ8X4 11249540 Ki = 3.8 nM T02551 C7BG9T 11258233 Ki = 2.5 nM T02551 C7XI0R 11260032 Ki = 0.631 nM T02551 CC0YP2 11271099 Ki = 0.1995 nM T02551 CL0DP6 11272440 Ki = 0.2512 nM T02551 CVO64A 11277053 Ki = 2089.3 nM T02551 C27GXZ 11277680 IC50 > 10000 nM T02551 CUJ2R7 11280344 Ki = 52.5 nM T02551 CZG20K 11281627 Ki = 1 nM T02551 C48WZU 11282073 Ki = 1.3 nM T02551 CDHK45 11290046 Ki = 22.91 nM T02551 CC2Y4X 11299620 Ki = 0.54 nM T02551 C57GTA 11299968 IC50 > 10000 nM T02551 C9BLC7 11304596 Ki = 199.53 nM T02551 CJS9C0 11304851 IC50 > 3200 nM T02551 CIMB79 11305766 Ki = 0.5012 nM T02551 C4DSN3 11307083 Ki = 3.4 nM T02551 CUXZ91 11311148 IC50 > 10000 nM T02551 C2GZD3 11311204 IC50 > 10000 nM T02551 CZ8M3K 11311583 Ki = 48.98 nM T02551 CU2GF6 11316078 Ki = 2 nM T02551 CXC2R6 11316847 Ki = 0.7 nM T02551 C6FD1Z 11317018 Ki = 3.8 nM T02551 CD03UE 11324141 Ki = 25 nM T02551 CH35RX 11327651 Ki = 1.2 nM T02551 CTIX74 11338096 Ki = 3760 nM T02551 CRMK35 11338674 Ki = 2 nM T02551 C2SQP0 11346463 Ki = 3630.78 nM T02551 CWR57Z 11346873 Ki = 4365.16 nM T02551 C0NRE8 11346967 Ki = 2408 nM T02551 CJT5E1 11350623 Ki = 31 nM T02551 CCY23Q 11351639 Ki = 1.1 nM T02551 CX7S0U 11352111 Ki = 0.9 nM T02551 CA1NC6 11356479 Ki = 6.7 nM T02551 C8D3CL 11357520 Ki = 4786.3 nM T02551 CXWH42 11358377 Ki > 10000 nM T02551 CDQ52C 11369049 Ki = 45.71 nM T02551 C82QCU 11375068 Ki = 0.9 nM T02551 CD5S7X 11380011 Ki = 2818.38 nM T02551 C4B3XN 11382976 Ki = 263.03 nM T02551 CBV52J 11384146 Ki = 930 nM T02551 C1OM3C 11384207 Ki = 1.698 nM T02551 C4SZ7W 11384664 Ki = 0.7 nM T02551 C9GP6C 11391402 Ki = 30.9 nM T02551 C6P2MT 11392229 Ki = 88.6 nM T02551 CQ5BN6 11396088 Ki = 1.7 nM T02551 C9AOM3 11397017 Ki = 1 nM T02551 CF4OX6 11397149 Ki = 31.62 nM T02551 C82ERW 11397777 Ki = 0.2512 nM T02551 C6MYE7 11403724 Ki = 2398.83 nM T02551 C1V4EQ 11404156 Ki > 10000 nM T02551 CDV4A0 11405107 Ki = 670 nM T02551 CT32OJ 11406143 Ki = 2860 nM T02551 C2ZCG3 11407062 Ki = 2.6 nM T02551 CGN10L 11408148 Ki = 2.1 nM T02551 C1XD0I 11408287 Ki = 3.4 nM T02551 C91RNU 11419120 Ki = 3 nM T02551 CKET16 11428547 Ki = 87.1 nM T02551 CO6F2D 11431895 Ki = 1.4 nM T02551 CW4O0K 11438733 Ki = 1548.82 nM T02551 C6S1FL 11442000 Ki = 2.6 nM T02551 CU3A2F 11442772 Ki = 0.3 nM T02551 CTM1W8 11443078 Ki = 0.5 nM T02551 C4PY8C 11450176 Ki = 1905.46 nM T02551 C86CJB 11451022 Ki = 45.1 nM T02551 C6SVK9 11452692 Ki = 2.4 nM T02551 C05VEA 11453253 Ki = 3.09 nM T02551 C8P0VE 11460104 Ki = 12022.64 nM T02551 CTA58W 11469395 Ki = 683 nM T02551 C8L6ZI 11472028 Ki > 10000 nM T02551 C3GMQ1 11477018 Ki = 0.7943 nM T02551 C4V1MG 11477201 Ki = 1.3 nM T02551 C2HU6O 11480902 Ki = 581 nM T02551 CFE98H 11487464 Ki = 2.7 nM T02551 C8BY4A 11489501 Ki > 501.19 nM T02551 C8FN2P 11494093 Ki = 73 nM T02551 COI68V 11496213 Ki = 41 nM T02551 CPX26I 11496746 Ki = 31.62 nM T02551 CNC9V7 11496793 Ki = 1140 nM T02551 C5Z7GQ 11497411 Ki = 2.512 nM T02551 C9YU1O 11497679 Ki = 5.012 nM T02551 CQT5U8 11497680 Ki = 3.981 nM T02551 C9JD4N 11497924 Ki = 79.43 nM T02551 CAU1R7 11500677 Ki = 150.5 nM T02551 CASD80 11501253 Ki > 1000 nM T02551 C16AXW 11501537 Ki = 214 nM T02551 C3ROH5 11504077 Ki = 0.7943 nM T02551 CN84HD 11504199 Ki = 19.3 nM T02551 CN63TR 11504230 Ki = 0.19 nM T02551 CXE65Q 11505572 Ki = 220 nM T02551 CRDF59 11509984 Ki = 77.9 nM T02551 C3TDJ2 11510684 Ki = 3.4 nM T02551 CF45XR 11511026 Ki = 0.6 nM T02551 COT4H9 11511117 Ki = 31.62 nM T02551 C9BT2W 11512263 Ki = 33.88 nM T02551 C7FH8P 11512962 Ki = 262 nM T02551 C59SCV 11516033 Ki = 1700 nM T02551 CAMP52 11517928 Ki = 850 nM T02551 C2MF1H 11518173 Ki = 6.9 nM T02551 CQ0IF2 11518499 Ki = 5539 nM T02551 CJ0B8E 11518546 Ki > 2700 nM T02551 CZ3D5Y 11518933 Ki = 63.1 nM T02551 C0WU7G 11518972 Ki = 12.59 nM T02551 CM4B3J 11519133 Ki = 7.943 nM T02551 C08JSL 11519134 Ki = 12.59 nM T02551 C04RCG 11519858 Ki = 12.59 nM T02551 CQ5IN9 11522339 Ki = 215 nM T02551 CO95XH 11525938 Ki = 3.162 nM T02551 CTNX29 11526451 Ki = 3.981 nM T02551 CR9NA7 11526531 Ki = 50.12 nM T02551 CNL15V 11527195 Ki = 50.12 nM T02551 C38QFE 11530118 IC50 > 10000 nM T02551 CPKR36 11533234 Ki = 10.6 nM T02551 CJF92G 11533429 Ki = 25.12 nM T02551 C2EQ1U 11533448 Ki = 15.85 nM T02551 C4LOQ9 11533473 Ki = 6.31 nM T02551 CZW9U3 11534726 Ki = 100 nM T02551 C2JT3I 11536995 Ki = 1833 nM T02551 C7DBO0 11537385 Ki = 144 nM T02551 CQ08DH 11539632 IC50 = 1.3 nM T02551 CSN91H 11539722 Ki = 31.62 nM T02551 C0X6CJ 11540474 Ki = 19.95 nM T02551 CO0R2G 11540842 Ki = 8.511 nM T02551 CN3W7S 11543350 Ki > 10000 nM T02551 C5ZY6N 11545813 Ki = 548.1 nM T02551 C7QKD5 11547151 Ki = 67.61 nM T02551 CD14OF 11547466 Ki = 39.81 nM T02551 CO5GF0 11547643 Ki = 102 nM T02551 C61LDE 11548217 Ki = 3.981 nM T02551 CKZ9B0 11548239 Ki = 1.995 nM T02551 CPA7K8 11548755 Ki = 63.1 nM T02551 C9VC7O 11551780 IC50 > 10000 nM T02551 C0ZBJ6 11554490 Ki = 1 nM T02551 C9XJP4 11554548 Ki = 10 nM T02551 CHDO61 11554831 Ki = 127 nM T02551 CBD05S 11554891 Ki = 85 nM T02551 C0VMG7 11555265 Ki = 1.585 nM T02551 C3Y4GR 11555971 Ki = 5.012 nM T02551 C7S2WZ 11558055 Ki = 47 nM T02551 C1V5CH 11559090 Ki > 10000 nM T02551 CY5I0U 11559581 Ki = 7700 nM T02551 CH67TN 11560697 Ki = 190 nM T02551 C4N0JC 11561601 Ki = 3.162 nM T02551 CX1VD8 11562113 Ki = 25.12 nM T02551 C0JU9T 11562199 Ki = 2.512 nM T02551 C4N8JS 11562200 Ki = 19.95 nM T02551 CVP1Q9 11567578 Ki = 5 nM T02551 CEV2P7 11567620 Ki = 309 nM T02551 CD3Z7J 11567928 Ki = 9.4 nM T02551 CG7VZ5 11568232 Ki = 4.23 nM T02551 CUH8Y7 11568543 Ki > 8500 nM T02551 C52PDV 11568714 Ki = 79.43 nM T02551 CR7M5S 11568725 Ki = 184 nM T02551 CNH1K4 11568826 Ki = 1.18 nM T02551 C0V5IK 11569099 Ki = 22.6 nM T02551 CCO29B 11569488 Ki = 38 nM T02551 C5J2UP 11569619 Ki = 4.266 nM T02551 CU6EY8 11569996 Ki = 2.512 nM T02551 CRK97Z 11570471 Ki = 3.467 nM T02551 C32JGN 11570589 Ki = 7.413 nM T02551 CP8MF4 11573628 Ki = 27.7 nM T02551 C1TBC8 11573806 Ki = 101.5 nM T02551 CTG5X1 11574902 Ki = 800 nM T02551 C8NMI4 11575479 Ki > 10000 nM T02551 C1Q8LC 11575799 Ki = 1000 nM T02551 C84MJZ 11576059 Ki = 12.59 nM T02551 CASH81 11576387 Ki = 3.981 nM T02551 CE60FY 11576528 Ki = 15.85 nM T02551 C8YLD3 11577158 Ki = 31.62 nM T02551 CZEB03 11577696 Ki = 23.9 nM T02551 CR8E2F 11578028 Ki = 100 nM T02551 C6JC2T 11580039 IC50 > 10000 nM T02551 C8CU1X 11581237 Ki = 1400 nM T02551 C4BGF8 11581443 Ki = 7.8 nM T02551 CQ09NJ 11583188 Ki = 600 nM T02551 C0HFP7 11584185 Ki = 7.943 nM T02551 CS1OR8 11584530 Ki = 194 nM T02551 C6D1MA 11584660 Ki = 1 nM T02551 CU4J2W 11584694 Ki = 7.943 nM T02551 CI2FK6 11584858 Ki = 15.14 nM T02551 CN5DQ9 11585034 Ki = 25.12 nM T02551 C73UHS 11585248 Ki = 39.81 nM T02551 C3V6LN 11590801 Ki = 53 nM T02551 CC75MD 11590828 Ki = 10 nM T02551 CYX50J 11591601 Ki = 25.12 nM T02551 CIUL60 11591633 Ki = 7.943 nM T02551 CU45DK 11595209 Ki > 10000 nM T02551 C5Q8XM 11595240 Ki = 1.88 nM T02551 C5NRD9 11596521 Ki = 0.54 nM T02551 CQ4SL7 11596603 Ki = 11.9 nM T02551 C1TOP5 11598123 Ki = 12.59 nM T02551 C6G7WS 11603119 Ki = 200 nM T02551 CGD62Y 11603486 Ki = 41 nM T02551 CU2V5R 11603959 Ki = 14.7 nM T02551 C9L3NI 11605088 Ki = 21.4 nM T02551 C9DI6R 11606176 Ki = 1 nM T02551 CO1A5Z 11606378 Ki = 1.995 nM T02551 CL04ZJ 11606435 Ki = 50.12 nM T02551 CJC5N8 11606456 Ki = 39.81 nM T02551 CZPE61 11608015 Ki = 2220 nM T02551 C2AFI7 11611862 Ki = 25.5 nM T02551 C9VOB8 11613105 Ki = 87.1 nM T02551 CT16JP 11613587 Ki = 3.162 nM T02551 CN91SZ 11613873 Ki = 39.81 nM T02551 C9BZG0 11615489 EC50 = 3.4 nM T02551 C62SOL 11615782 Ki > 4000 nM T02551 C7XB8E 11618408 Ki = 4.7 nM T02551 CKB59U 11620847 Ki = 25.12 nM T02551 CXY07A 11621352 Ki = 1 nM T02551 CN1P4I 11623343 Ki = 342 nM T02551 CB7M8E 11625642 Ki = 8.8 nM T02551 CC2G9I 11626748 Ki = 880 nM T02551 C9FSA8 11627847 Ki = 3.162 nM T02551 C51IBH 11627879 Ki = 39.81 nM T02551 CE8W1Z 11628452 Ki = 7.943 nM T02551 CFJN71 11628631 Ki = 5.012 nM T02551 C8R6MK 11630058 Ki = 12000 nM T02551 C8ZU2X 11631892 Ki = 3500 nM T02551 C7CZE3 11633170 Ki = 2100 nM T02551 CMZR85 11633816 Ki = 5.2 nM T02551 C5W0JR 11633992 Ki = 2431 nM T02551 CG1C3D 11637457 Ki = 87 nM T02551 C2OU7Y 11638332 Ki > 10000 nM T02551 C19UMY 11638640 Ki = 62 nM T02551 CI17EA 11638780 Ki = 5600 nM T02551 CH89AK 11639248 Ki = 55 nM T02551 C0XC2N 11641596 Ki = 50.12 nM T02551 C25KGE 11641641 Ki = 3.162 nM T02551 C8DXS0 11642163 Ki = 5.012 nM T02551 CEN25S 11646648 Ki = 580 nM T02551 CMIC92 11647002 Ki = 895 nM T02551 CZX78K 11647384 Ki = 32.6 nM T02551 CYQB50 11648990 Ki = 19.95 nM T02551 C9XD0H 11649431 Ki = 2.399 nM T02551 CEZO71 11652518 Ki = 60000 nM T02551 C1HDM5 11653679 Ki = 158.8 nM T02551 C2R9QT 11654739 Ki = 0.27 nM T02551 CJV2I4 11655403 Ki = 143 nM T02551 C5T4UV 11655570 Ki = 470 nM T02551 C48HCV 11656243 Ki = 63.1 nM T02551 CPE83G 11656848 Ki = 6.31 nM T02551 CT14BC 11657494 Ki = 19.95 nM T02551 CP21DV 11658914 EC50 = 4.5 nM T02551 C7NHO6 11659604 Ki = 42000 nM T02551 CD79UX 11661609 Ki = 670 nM T02551 CEL15N 11662194 Ki = 100 nM T02551 C6R1GA 11662426 Ki = 118 nM T02551 C4L7TV 11662592 Ki = 1.3 nM T02551 CBU0L8 11663504 Ki = 39.81 nM T02551 C69RQX 11663526 Ki = 19.95 nM T02551 C3SJO5 11663578 Ki = 25.12 nM T02551 CO2HB4 11663604 Ki = 12.88 nM T02551 C1PB0O 11663999 Ki = 1.585 nM T02551 C16UWH 11664328 Ki = 39.81 nM T02551 C6URZ0 11668565 Ki = 122 nM T02551 CNE2K5 11669953 Ki = 63.1 nM T02551 CY0J2U 11670421 Ki = 28.84 nM T02551 CQR15M 11670438 Ki = 1440 nM T02551 C2EUR0 11671211 Ki > 8500 nM T02551 CGXE47 11672839 Ki = 1520 nM T02551 CH8M9X 11673558 Ki = 17000 nM T02551 CH9M7J 11675867 IC50 = 0.7 nM T02551 CY4B9F 11676195 Ki = 0.35 nM T02551 CY5UB8 11676600 Ki = 8.6 nM T02551 C4KUL7 11676638 Ki = 0.2 nM T02551 CMQX39 11676873 Ki = 0.3 nM T02551 CWQ3M4 11677768 Ki = 3.981 nM T02551 C6C4BJ 11678080 Ki = 15.85 nM T02551 CTK8R9 11678172 Ki = 0.46 nM T02551 CSQ4B1 11681599 Ki = 24.6 nM T02551 CVRW29 11682812 Ki = 2400 nM T02551 C1ZD6V 11685267 Ki = 12.59 nM T02551 CS1WO0 11689612 Ki = 1000 nM T02551 CRM26C 11691676 Ki = 1285 nM T02551 CG13YQ 11691697 Ki = 1.585 nM T02551 C5J7PY 11692038 Ki = 98 nM T02551 CE1KI3 11692214 Ki = 31.62 nM T02551 CGM36K 11692376 Ki = 25.12 nM T02551 C3LYZ6 11694483 Ki = 12000 nM T02551 CDV58J 11696813 Ki = 4.5 nM T02551 C1W8NR 11696910 Ki = 1500 nM T02551 C9ED1Y 11697270 Ki = 390 nM T02551 CT5J9M 11699340 Ki = 6.31 nM T02551 CB4H2O 11699469 Ki = 16 nM T02551 C2YE9V 11699516 Ki = 32.36 nM T02551 CFCB20 11699532 Ki = 0.7943 nM T02551 CUY90O 11704609 Ki = 3.7 nM T02551 CGD80W 11705119 Ki = 12.59 nM T02551 C2E8BF 11705395 Ki = 3.1 nM T02551 CLK68A 11705570 Ki = 5.012 nM T02551 CPC67X 11705929 Ki = 1.995 nM T02551 CJL61W 11706497 Ki = 3.6 nM T02551 C3EP0X 11708363 Ki = 2100 nM T02551 CL08TQ 11711943 Ki = 2322 nM T02551 CN8FE3 11712044 Ki = 100 nM T02551 C5RZ3S 11712530 Ki = 0.105 nM T02551 CZ6NB8 11716438 Ki = 296 nM T02551 C9FTL5 11718008 Ki = 415 nM T02551 C7T1IL 11720119 Ki = 10.96 nM T02551 CGO56C 11720302 Ki = 1.9 nM T02551 CI1W3L 11720433 Ki = 93.8 nM T02551 CXUM63 11720838 Ki = 0.7943 nM T02551 C37DMH 11721190 Ki = 3.981 nM T02551 CXYQ40 11725531 Ki = 26000 nM T02551 CNPU72 11725909 Ki = 900 nM T02551 CVL96I 11729782 Ki = 3.3 nM T02551 C7UA6T 11730189 Ki = 6.7 nM T02551 C7PVL8 11730467 IC50 = 758 nM T02551 C1JKS2 11731962 Ki = 0.33 nM T02551 C8L0KE 11732280 Ki = 15.5 nM T02551 C50XKE 11733317 Ki = 750 nM T02551 C2B7EY 11733372 Ki = 16 nM T02551 C15MBU 11736707 Ki = 2818.38 nM T02551 C0URA1 11740275 Ki = 10 nM T02551 CJIB79 11742742 Ki = 316.23 nM T02551 CQP6N4 11743225 Ki = 0.7943 nM T02551 CPG15O 11743399 IC50 > 1000 nM T02551 CYV02C 11747350 Ki = 110 nM T02551 CG0YB2 11751828 Ki = 1 nM T02551 C5L2TO 11754850 Ki = 4.8 nM T02551 CD4Q5T 11761090 Ki = 4.8 nM T02551 C1MQ6G 11761374 Ki = 1 nM T02551 C5EH3J 11761412 Ki = 0.34 nM T02551 CQX0T6 11762743 Ki = 36 nM T02551 C0KZ3P 11767026 Ki = 14.9 nM T02551 CZGB28 11770929 Ki = 6025.6 nM T02551 CV3OA5 11774865 Ki = 0.6 nM T02551 C5QGC3 11775544 Ki = 1.585 nM T02551 CB46KD 11776309 EC50 > 10000 nM T02551 CV91RG 11778580 Ki = 1384 nM T02551 CK4IQ8 11778702 Ki = 78 nM T02551 C3RAX7 11784937 Ki = 3.15 nM T02551 CT8LD5 11792163 Ki > 3030 nM T02551 CAQP08 11792373 Ki > 3030 nM T02551 CHQ38Z 11794122 Ki = 24 nM T02551 CEW12K 11794570 Ki = 430 nM T02551 CJA41D 11795011 Ki = 11 nM T02551 CN9M8E 11811722 IC50 = 149 nM T02551 CWMA41 11812065 Ki = 4.1 nM T02551 CO5Y7T 11812299 Ki = 29 nM T02551 CGFW41 11812838 Ki = 24 nM T02551 CWFC60 11812905 Ki = 10.1 nM T02551 C6IWM9 11826097 Ki = 0.46 nM T02551 CSNC92 11826347 Ki = 325 nM T02551 CJ1UD5 11826673 Ki = 2.14 nM T02551 CXLW54 11948707 Ki > 10000 nM T02551 C23IVY 11957566 EC50 = 0.95 nM T02551 CPKV28 11957618 IC50 = 80 nM T02551 C7RY5S 11983282 EC50 = 3.3 nM T02551 CR4YS2 11996303 Ki = 0.7943 nM T02551 C7D1AY 11996304 Ki = 0.631 nM T02551 C02JVQ 12049520 Ki = 3950 nM T02551 CXTH25 12049521 Ki = 660 nM T02551 C9V1XN 12049907 Ki = 25.12 nM T02551 C1U7RH 12049908 Ki = 19.95 nM T02551 C37GTL 12049910 Ki = 6.31 nM T02551 CVN2P5 12049911 Ki = 6.31 nM T02551 C57VXR 12050193 Ki = 1190 nM T02551 CV56XD 12050194 Ki = 8400 nM T02551 C5C2GB 12050195 Ki = 1050 nM T02551 C64JUP 12050196 Ki = 5250 nM T02551 C4QHA5 12050197 Ki = 640 nM T02551 CAL98J 12050198 Ki = 6100 nM T02551 CJ7W9T 12050199 Ki = 580 nM T02551 CXEV76 12050200 Ki = 2300 nM T02551 CP5W7X 12050201 Ki = 205 nM T02551 CZHQ31 12050202 Ki = 1700 nM T02551 CX47WZ 12052258 Ki = 120 nM T02551 C6QEW2 12066264 Ki = 112 nM T02551 CF4D5H 12066265 Ki = 277 nM T02551 C9G7LR 12071089 Ki = 72.7 nM T02551 CT8SE7 12280575 Ki = 529 nM T02551 CHQ45V 12280580 Ki = 76 nM T02551 C4NWX9 12301195 Ki > 10000 nM T02551 C1QYW7 12461787 Ki = 21542 nM T02551 CS3JE5 12581154 Ki = 409 nM T02551 C9XLS6 12581156 Ki = 501 nM T02551 C72ZLP 12581164 Ki = 603 nM T02551 CU3XH9 12581203 Ki = 857 nM T02551 CEBK96 12581219 Ki = 361 nM T02551 CK1X6Z 12741429 Ki = 366 nM T02551 CZT58X 12888943 Ki = 160 nM T02551 CNW1I4 12898419 Ki = 36 nM T02551 C8ON5D 12899499 Ki = 7.4 nM T02551 CPY6L8 12899569 Ki = 5.7 nM T02551 C5MB7I 12997400 Ki = 570 nM T02551 CXM15G 12997412 Ki = 430 nM T02551 CP0MN1 12997413 Ki = 170 nM T02551 C2V9FL 13091268 Ki = 0.7079 nM T02551 CCG14E 13091356 Ki = 4.1 nM T02551 C1JW2Q 13091358 Ki = 4.1 nM T02551 CYN95Z 13091359 Ki = 0.7 nM T02551 CC74ND 13373172 Ki = 306.5 nM T02551 CJ75SB 13670706 Ki = 1.9 nM T02551 C86GDA 13680883 Ki > 100000 nM T02551 C39SGZ 13687192 Ki = 28 nM T02551 C1H9QW 13767784 Ki = 6.2 nM T02551 C14SUX 13805900 Ki = 0.54 nM T02551 CWS14H 13869641 Ki = 41 nM T02551 C3Z4DN 14465382 EC50 = 0.73 nM T02551 CV52EC 14601425 Ki = 0.16 nM T02551 CSM29P 14665503 Ki = 0.6 nM T02551 CMO81H 14925759 Ki = 1318.26 nM T02551 CC47XA 14973078 Ki = 273 nM T02551 CY4E2W 14977566 Ki = 691 nM T02551 CZB32N 15006482 EC50 > 1000 nM T02551 C5MJ2V 15006484 EC50 > 2800 nM T02551 CDM02J 15006491 EC50 = 27 nM T02551 C5W4MG 15034333 Ki > 5000 nM T02551 CL7P9W 15045455 Ki = 4.3 nM T02551 C6R7OW 15232471 Ki = 79.43 nM T02551 CWJ2L5 15232472 Ki = 76 nM T02551 C5G3LK 15232474 Ki = 63.1 nM T02551 C36JOH 15232475 Ki = 50 nM T02551 CNP2K1 15232476 Ki = 39 nM T02551 CV7ZG5 15232477 EC50 = 28 nM T02551 CW52NY 15232478 Ki = 132 nM T02551 C0VYU7 15232479 Ki = 50.12 nM T02551 CLXP32 15232480 Ki = 79.43 nM T02551 CMS94O 15232481 Ki = 79.43 nM T02551 C04JQR 15232482 Ki = 131 nM T02551 CUI42N 15291583 Ki = 9 nM T02551 C6CO3J 15291585 Ki = 133 nM T02551 C76GUO 15291586 Ki = 184 nM T02551 CQ30UI 15291587 Ki = 35 nM T02551 C13GNK 15293841 Ki = 403 nM T02551 CJIS26 15356306 Ki = 54.6 nM T02551 CH6A1U 15388745 Ki = 0.5 nM T02551 CDV47F 15389744 Ki > 10000 nM T02551 CGD3K7 15389746 Ki > 10000 nM T02551 CGZ5A0 15389747 Ki = 2754.23 nM T02551 CIAB49 15389749 Ki = 2630.27 nM T02551 CF6HQ7 15431693 Ki = 1.4 nM T02551 C4KNM7 15467369 Ki = 5250 nM T02551 C5UO3R 15467370 Ki = 31000 nM T02551 CCB94N 15467371 Ki = 6950 nM T02551 C2B0NM 15467372 Ki = 6950 nM T02551 CCMQ75 15467373 Ki = 7600 nM T02551 C5FWQ2 15508238 Ki = 8700 nM T02551 C8VB3H 15508239 Ki = 7700 nM T02551 C5NC6J 15508242 Ki = 31000 nM T02551 C30CHU 15512229 Ki < 316.23 nM T02551 C15PZT 15522515 Ki = 1600 nM T02551 CW50JX 15651970 Ki = 1372 nM T02551 CK5P6M 15651971 Ki = 3055 nM T02551 C59WZE 15654433 Ki = 68 nM T02551 C12WNY 15654434 Ki > 1623 nM T02551 C0VAS7 15720219 Ki = 575.44 nM T02551 CLN26K 15720220 Ki = 560 nM T02551 CUE15H 15817167 Ki = 27 nM T02551 CXG2S4 15817168 Ki = 130 nM T02551 C81RSY 15817169 Ki = 155 nM T02551 CTPS81 15817172 Ki = 8 nM T02551 CD30XV 15840855 IC50 = 150 nM T02551 CW9M5X 15888352 Ki > 3000 nM T02551 C74UVA 15937765 EC50 = 1890 nM T02551 C0HAO3 15949564 Ki = 0.8 nM T02551 C9CGE4 16007814 Ki = 1900 nM T02551 CG4KC8 16038360 EC50 = 1.03 nM T02551 CAUP23 16048564 Ki = 330 nM T02551 CWMC70 16090814 Ki = 277.5 nM T02551 CP09RQ 16090821 Ki = 521 nM T02551 C5Q8DR 16094666 Ki = 433 nM T02551 CS1D0G 16121920 Ki = 6100 nM T02551 CYV05C 16123136 Ki = 2.512 nM T02551 C8C2IW 16123138 Ki = 2.512 nM T02551 C7YF8I 16123140 Ki = 7.943 nM T02551 C91DQN 16123241 Ki = 6.31 nM T02551 CQG7P8 16123247 Ki = 1.259 nM T02551 CA6D4S 16123347 Ki = 25.12 nM T02551 CBH5P4 16123349 Ki = 251.19 nM T02551 CPN48R 16123353 Ki = 5.012 nM T02551 CK7H2W 16123462 Ki = 6.31 nM T02551 C5MY2Q 16123464 Ki = 630.96 nM T02551 CNQ6J2 16123467 Ki = 25.12 nM T02551 CZ2IS9 16660294 Ki > 10000 nM T02551 CGX0D5 16665071 Ki = 3.78 nM T02551 CRIH69 16744003 Ki = 5.1 nM T02551 C3D0FE 16744004 Ki = 2.1 nM T02551 CKDM79 16744005 Ki = 20 nM T02551 CQ1MG0 16744171 Ki = 2.1 nM T02551 CTI89R 16759249 Ki = 34.4 nM T02551 CHLR19 17424979 EC50 = 3300 nM T02551 C8ZK9L 17440212 EC50 = 430 nM T02551 CF25CM 17449900 EC50 = 0.21 nM T02551 C73MFP 17469721 Ki = 2900 nM T02551 CPZJ30 17475863 Ki = 537.03 nM T02551 C7KP5T 17755866 Ki = 6122 nM T02551 CX7VE8 17755867 Ki = 100 nM T02551 CUW8S4 17755868 Ki = 3964 nM T02551 C3KA6Z 17755875 Ki > 10000 nM T02551 C4N1LS 17755991 Ki = 6896 nM T02551 C6BE2Y 17755992 Ki > 10000 nM T02551 C10UQJ 17755999 Ki = 3136 nM T02551 C6WO9X 17756101 Ki = 507 nM T02551 CI9RW0 17756102 Ki = 1349 nM T02551 CDPT42 17756110 Ki > 10000 nM T02551 C0XG9B 17756212 Ki = 23903 nM T02551 C6JQ1K 17756213 Ki = 776 nM T02551 CTF31I 17866220 Ki = 3.981 nM T02551 CG69RD 17866221 Ki = 3.981 nM T02551 CR3A2X 17866228 Ki = 5.012 nM T02551 CZR2T6 17866229 Ki = 3.981 nM T02551 CV4N5L 17866237 Ki = 3.162 nM T02551 CP4YQ5 17866241 Ki = 3.981 nM T02551 C8D3RM 17866242 Ki = 3.981 nM T02551 C2ATF6 17866249 Ki = 3.981 nM T02551 CU9XT8 17867623 Ki = 0.7943 nM T02551 CPQR14 17867626 Ki = 1.585 nM T02551 CL5C3X 17888044 IC50 = 200 nM T02551 C87POY 17895586 Ki = 2.512 nM T02551 C3HO5U 17895587 Ki = 1.995 nM T02551 CZ78BE 17987129 Ki > 4200 nM T02551 C9PV8A 18180076 IC50 = 2102 nM T02551 CMQT08 18397434 Ki > 10000 nM T02551 C9DQU7 18414156 Ki = 56.5 nM T02551 CUW96J 18596256 Ki = 1 nM T02551 CJ20BQ 18624462 Ki = 21 nM T02551 CW04FC 18702006 Ki = 7.943 nM T02551 CS5QC2 18702007 Ki = 12.59 nM T02551 CYI8L6 18702008 Ki = 1 nM T02551 CLK87H 18706871 Ki = 10 nM T02551 CGTJ59 18715674 Ki = 6.31 nM T02551 C3M6CU 18715682 Ki = 15.85 nM T02551 CPSI76 18797033 Ki = 2.512 nM T02551 C91OCW 18797049 Ki = 7.943 nM T02551 CWXR15 18993044 Ki = 15 nM T02551 CU8TB3 19041559 Ki = 56 nM T02551 CREN73 19043055 Ki = 5.012 nM T02551 C0MY7J 19043056 Ki = 0.7943 nM T02551 C0MB8I 19370371 Ki = 500 nM T02551 C6AOE8 19426635 IC50 = 338.84 nM T02551 CJ7RL6 19592091 Ki = 0.1995 nM T02551 CT08UM 19592101 Ki = 12.59 nM T02551 C70DZN 19592119 Ki = 2.512 nM T02551 CG47ID 19592121 Ki = 0.7943 nM T02551 C09EYA 19592126 Ki = 1.259 nM T02551 CO3QN2 19592133 Ki = 1.585 nM T02551 C8E3FM 19592141 Ki = 3.981 nM T02551 CMC12O 19592159 Ki = 0.5012 nM T02551 CRF1H4 19608536 Ki = 4.7 nM T02551 CW61QX 19694408 Ki = 79.43 nM T02551 CQN56J 19694436 Ki = 15.85 nM T02551 CCZ04S 19694443 Ki = 79.43 nM T02551 C10BRS 19694446 Ki = 15.85 nM T02551 CYJ3Z4 19694453 Ki = 125.89 nM T02551 C1JTW4 19871273 Ki = 36.3 nM T02551 C61OBX 19881394 Ki = 1098 nM T02551 C43ACN 19938402 Ki = 144 nM T02551 C1PS8O 19938405 Ki = 26 nM T02551 CC8A3Z 19938408 Ki = 8 nM T02551 CEN3L5 19964401 Ki = 3210 nM T02551 C5IHG3 19964406 Ki = 10800 nM T02551 C9VXS1 19964410 Ki = 1480 nM T02551 CG8Z4W 20256387 Ki > 400 nM T02551 C3DQS5 20267107 Ki = 1566 nM T02551 CB0NH7 20267108 Ki = 83 nM T02551 C56JNM 21085427 Ki = 149 nM T02551 CP2R7D 21186098 IC50 = 320 nM T02551 CNR17B 21186102 IC50 = 72 nM T02551 CXY0P4 21186115 IC50 = 8 nM T02551 CY0QO4 21186124 IC50 = 33 nM T02551 C79MJX 21186138 IC50 = 300 nM T02551 CUJ4R9 21186143 IC50 = 1100 nM T02551 CGY9F6 21186148 IC50 = 480 nM T02551 CRA23J 21186186 IC50 = 59 nM T02551 C18IWL 21186192 IC50 = 200 nM T02551 C5ER6Q 21186194 IC50 = 710 nM T02551 CLN86H 21219144 Ki = 1400 nM T02551 C2M0HK 21219154 Ki = 810 nM T02551 C1GQY9 21219156 Ki = 2200 nM T02551 C6LM2O 21219157 Ki = 28 nM T02551 C0W8PE 21219160 Ki = 1300 nM T02551 CG4XF7 21219164 Ki = 820 nM T02551 C9S5XI 21219166 Ki = 740 nM T02551 CH83US 21219167 Ki = 2500 nM T02551 C60TBU 21219173 Ki > 4400 nM T02551 CB3KF6 21219176 Ki = 260 nM T02551 C94BPG 21460314 Ki = 0.9 nM T02551 C7MYT1 21462964 Ki = 1300 nM T02551 C8GC6E 21462980 Ki = 170 nM T02551 C2D6ZX 21465540 Ki > 4400 nM T02551 C3T5HF 21509921 Ki > 10000 nM T02551 CFN81Q 21527771 Ki = 49 nM T02551 CH59WN 21533446 Ki = 49 nM T02551 CRE80D 21559988 Ki = 1700 nM T02551 CAH39X 21564536 Ki > 10000 nM T02551 CT7XG9 21830793 Ki > 10000 nM T02551 CG08FZ 21969199 Ki = 15.85 nM T02551 C0EGL8 21969201 Ki = 1.995 nM T02551 C4TQ5H 21969204 Ki = 5.012 nM T02551 C20AOH 21969205 Ki = 7.943 nM T02551 CMH48V 21973550 Ki = 1.995 nM T02551 CLF09T 22065962 Ki = 1500 nM T02551 CYCS06 22100932 Ki = 660 nM T02551 CM75DA 22100933 Ki = 2900 nM T02551 CP48JW 22100940 Ki = 560 nM T02551 C68MQE 22100943 Ki = 630 nM T02551 CWH1R0 22100957 Ki > 4500 nM T02551 C9TG8S 22100962 Ki = 1800 nM T02551 CLCN93 22100964 Ki = 1600 nM T02551 CC3LF7 22100965 Ki = 1400 nM T02551 C90FER 22100968 Ki = 4500 nM T02551 C9RUA4 22100970 Ki = 1600 nM T02551 C4SXJ3 22132503 Ki = 3.981 nM T02551 CS62AZ 22261332 Ki = 0.74 nM T02551 C2M4SX 22261340 Ki = 3.59 nM T02551 C0FTG5 22376257 Ki = 15.85 nM T02551 C9U1GM 22403029 Ki = 1.995 nM T02551 CGVE83 22403039 Ki = 1.995 nM T02551 C9KI2W 22403044 Ki = 63.1 nM T02551 C3FEL1 22403055 Ki = 39.81 nM T02551 CUNF84 22403068 Ki = 15.85 nM T02551 CM6YV2 22403070 Ki = 0.2512 nM T02551 CY0ZF7 22403109 Ki = 25.12 nM T02551 CCZ3U1 22403110 Ki = 19.95 nM T02551 C3GWZ7 22403137 Ki = 0.3162 nM T02551 CCZ5Q3 22622605 Ki = 3.981 nM T02551 CVX19H 22727322 Ki = 24 nM T02551 CT45YC 22727323 Ki = 6 nM T02551 CL26HS 22727324 Ki = 23 nM T02551 CCS83F 22727331 Ki = 6.5 nM T02551 CS5J2U 22727332 Ki = 10 nM T02551 CAUK40 22727334 Ki = 18 nM T02551 CSCJ35 22727335 Ki = 9.5 nM T02551 CCIW17 22727346 Ki = 38 nM T02551 CS9IF2 22727347 Ki = 15 nM T02551 CFQ92N 22727351 Ki = 60 nM T02551 CE2P3H 22727356 Ki = 27 nM T02551 C64UKQ 22727358 Ki = 15 nM T02551 CU6B2Z 22727361 Ki = 16 nM T02551 C4S2NC 22876327 Ki = 2.512 nM T02551 CAM3H4 22910005 Ki = 8.4 nM T02551 C8C3VU 23025506 Ki > 100000 nM T02551 C8IN9H 23202795 Ki = 1.259 nM T02551 C16PUX 23202799 Ki = 1.585 nM T02551 CVAB38 23202826 Ki = 1 nM T02551 C89NDA 23277137 Ki = 0.21 nM T02551 CEP65L 23364995 Ki = 56 nM T02551 CQSF94 23625084 Ki = 176 nM T02551 C5WOV6 23625240 Ki = 28.9 nM T02551 CNAK80 23625241 Ki = 8 nM T02551 CVRW14 23625242 Ki = 225 nM T02551 C4K8QX 23625243 Ki = 146 nM T02551 CPR07Q 23625244 Ki = 8 nM T02551 C43MPJ 23625385 Ki = 60 nM T02551 CRB85L 23625386 Ki = 54.4 nM T02551 CS0VM3 23625539 Ki = 156 nM T02551 CD7AK1 23625540 Ki = 71 nM T02551 C85WQO 23625541 Ki = 50 nM T02551 CESF95 23625542 Ki = 38 nM T02551 C9Z1EM 23625543 Ki = 40 nM T02551 CU0F6C 23625706 Ki = 385 nM T02551 CXD3E6 23625925 Ki = 186.21 nM T02551 CK6B7G 23630497 Ki = 1.259 nM T02551 CH95VG 23630499 Ki = 2.512 nM T02551 C2XLN1 23630501 Ki = 1 nM T02551 C1N5TV 23630503 Ki = 39.81 nM T02551 C7WZJ0 23630505 Ki = 10 nM T02551 C4MI9Y 23630602 Ki = 1.259 nM T02551 C24TDZ 23630604 Ki = 3.162 nM T02551 CU8D0O 23630606 Ki = 0.3981 nM T02551 CKB1E5 23630796 Ki = 1.995 nM T02551 CJ81PU 23630797 Ki = 3.162 nM T02551 CV68XN 23630900 Ki = 1.585 nM T02551 CD61SO 23630901 Ki = 1.585 nM T02551 CY2RG1 23630902 Ki = 1.995 nM T02551 CJ90YG 23630903 Ki = 1 nM T02551 CTJS17 23630998 Ki = 6.31 nM T02551 CXVR30 23630999 Ki = 1.585 nM T02551 CSAT45 23631000 Ki = 3.162 nM T02551 C6EO1W 23631001 Ki = 2.512 nM T02551 CE3AM4 23631091 Ki = 0.7943 nM T02551 C9BMW2 23631092 Ki = 1.585 nM T02551 CKT7B3 23631093 Ki = 5.012 nM T02551 CM8U1D 23631172 Ki = 1.259 nM T02551 CWZT34 23631173 Ki = 0.7943 nM T02551 CH2I1P 23631366 Ki = 1.585 nM T02551 C6YS4P 23631368 Ki = 25.12 nM T02551 C4TV8X 23631454 Ki = 0.631 nM T02551 CE40PT 23631458 Ki = 10 nM T02551 C09NTA 23631540 Ki = 1.995 nM T02551 C83QKW 23631544 Ki = 2.512 nM T02551 C0RPW8 23631636 Ki = 3.981 nM T02551 CI4B6N 23642427 Ki = 0.46 nM T02551 CO4C6M 23653115 Ki = 306 nM T02551 CBUJ02 23653176 Ki = 1204 nM T02551 C2BO0F 23928184 Ki = 58 nM T02551 CDH38J 23992579 Ki = 427 nM T02551 C3RS6J 24742011 EC50 = 0.12 nM T02551 C7BCW8 24754330 Ki = 22.2 nM T02551 C9SP0R 24754332 Ki = 10.9 nM T02551 C20IKD 24754400 EC50 = 0.08 nM T02551 CP0VE5 24754476 Ki = 0.45 nM T02551 CFEP49 24754538 Ki = 10.3 nM T02551 C5GYO8 24754540 Ki = 2.89 nM T02551 CYGH43 24754542 Ki = 0.825 nM T02551 C2XAQ7 24754913 Ki = 11.2 nM T02551 C39ZCR 24754914 Ki = 23.9 nM T02551 CWA40O 24754983 Ki = 1.39 nM T02551 CJ1QB7 24758481 Ki = 31.62 nM T02551 C8CWX4 24758715 Ki = 2.512 nM T02551 CU06GI 24758717 Ki = 7.943 nM T02551 CPL05Y 24758828 Ki = 7.943 nM T02551 C7RZ9I 24758830 Ki = 15.85 nM T02551 C6JQC4 24758832 Ki = 31.62 nM T02551 CBNF87 24758834 Ki = 100 nM T02551 CGQL10 24758836 Ki = 79.43 nM T02551 CGE32Q 24758838 Ki = 100 nM T02551 CL80CU 24758945 Ki = 50.12 nM T02551 C8JQW6 24758947 Ki = 31.62 nM T02551 CMB3J9 24759792 EC50 = 1.413 nM T02551 C6B1IG 24767784 Ki = 0.37 nM T02551 C0I2HU 24769156 Ki = 0.6 nM T02551 CP08DV 24805120 Ki = 891.25 nM T02551 CI15OJ 24805284 Ki = 19.05 nM T02551 C21VNW 24805285 EC50 = 4.677 nM T02551 CKW7R2 24805286 Ki = 120.23 nM T02551 CQ7S8N 24805287 EC50 = 2.291 nM T02551 C9K0CX 24805674 Ki = 15 nM T02551 C8TZY0 24810004 Ki = 63.3 nM T02551 CSCW01 24815434 Ki = 125.89 nM T02551 CBF6J9 24815439 Ki = 100 nM T02551 C0DYP7 24815883 Ki > 10000 nM T02551 CN9AY0 24815976 Ki > 10000 nM T02551 CYL30C 24823920 Ki = 590 nM T02551 CHC2B6 24823921 Ki = 410 nM T02551 C0Y8UL 24823922 Ki = 320 nM T02551 CB9Z8R 24824060 Ki = 3400 nM T02551 CTS57E 24824061 Ki = 930 nM T02551 C6ED9B 24824062 Ki = 940 nM T02551 CPT34W 24824063 Ki = 15000 nM T02551 CGU94D 24824065 Ki = 2200 nM T02551 C6Y4FV 24824066 Ki = 3400 nM T02551 C37MEX 24837518 EC50 = 667 nM T02551 CDC91N 24839550 Ki = 676.08 nM T02551 CY21RE 24841480 Ki = 1000 nM T02551 CF8I9P 24845776 Ki = 10 nM T02551 C1CUD0 24848444 Ki = 130 nM T02551 C2A0LT 24849462 Ki = 316.23 nM T02551 CBGO31 24867245 Ki = 1296 nM T02551 C1FZV4 24873453 Ki = 0.3 nM T02551 CKG9N0 24873454 Ki > 1000 nM T02551 C49GLI 24882561 Ki = 3900 nM T02551 C6L7KS 24887518 Ki = 457.09 nM T02551 CAOF91 24894071 IC50 > 10000 nM T02551 C69AYD 24900557 Ki = 199.53 nM T02551 C4IGH9 24936042 Ki = 20 nM T02551 CAP8R4 24936081 EC50 = 0.085 nM T02551 CTI38U 25060119 Ki = 3240 nM T02551 CD0YW2 25070416 Ki = 5.9 nM T02551 C5QU0F 25070419 Ki = 3.5 nM T02551 CTN36E 25070740 Ki = 10 nM T02551 CGAZ01 25070742 Ki = 20 nM T02551 CKB23A 25071066 Ki = 7 nM T02551 CI8NL3 25071384 EC50 = 1.9 nM T02551 C6F5SU 25071385 EC50 = 7.7 nM T02551 CL7TN4 25071691 Ki = 0.69 nM T02551 C75ZIC 25071692 Ki = 1.5 nM T02551 C49ZFU 25072002 Ki = 2.9 nM T02551 CM28GQ 25072632 Ki = 2.3 nM T02551 C8OBV4 25072633 Ki = 5 nM T02551 CIT6G4 25072635 Ki = 2 nM T02551 CS1CI4 25072941 Ki = 17 nM T02551 C3CLH5 25072943 Ki = 7.2 nM T02551 C1XSD0 25072946 Ki = 6.4 nM T02551 CBKG34 25093832 Ki = 3.3 nM T02551 C3W6DQ 25096873 Ki = 0.09 nM T02551 C9DZN4 25128753 Ki = 84.7 nM T02551 CT7U5K 25128755 Ki = 1210 nM T02551 C2FY7C 25128757 Ki = 3.62 nM T02551 CPZ7K5 25128759 Ki = 431 nM T02551 CL1HC0 25129111 Ki = 0.34 nM T02551 C8MX9U 25129113 Ki = 1.2 nM T02551 C2U0HS 25129115 Ki = 0.92 nM T02551 C0I8HD 25129458 Ki = 2 nM T02551 CTX43Q 25129459 Ki = 2.1 nM T02551 C6XMF9 25129460 Ki = 8.4 nM T02551 C5NW4M 25129807 IC50 = 12.3 nM T02551 C2O4KV 25129809 Ki = 31 nM T02551 CX3R5L 25130151 Ki = 541 nM T02551 CD2KY1 25130153 Ki = 21.2 nM T02551 C3I1FU 25130155 Ki = 17.9 nM T02551 CAV81B 25130157 Ki = 0.71 nM T02551 CRSZ60 25130159 Ki = 32.2 nM T02551 CIM1F4 25130509 Ki = 0.53 nM T02551 CFJ6Y9 25131876 Ki = 13.18 nM T02551 C67QCG 25132869 Ki = 6.35 nM T02551 CC0S6N 25132870 Ki = 480 nM T02551 CG9I6X 25132871 Ki = 224 nM T02551 C8Y5LD 25133211 Ki = 6410 nM T02551 CN61ZL 25139180 Ki = 300 nM T02551 CLTF40 25139181 Ki = 0.2 nM T02551 CN32VX 25139329 Ki = 150 nM T02551 C0LZ7B 25139335 Ki = 280 nM T02551 CW07GC 25139477 Ki = 4.4 nM T02551 CQD6N1 25139478 Ki = 13 nM T02551 CN3S7R 25139479 Ki = 1.3 nM T02551 CSG25V 25139481 Ki = 140 nM T02551 CXDM41 25141533 Ki = 1.8 nM T02551 CL84YJ 25141534 Ki = 1.39 nM T02551 C4FXR9 25141535 Ki = 1.4 nM T02551 CKBJ53 25141536 Ki = 7.71 nM T02551 C8OGB1 25141538 IC50 = 1.76 nM T02551 CX04LB 25142456 Ki = 390 nM T02551 CTIL36 25186021 Ki = 3.2 nM T02551 C0I3KU 25186022 Ki = 8.2 nM T02551 C52BNH 25186023 Ki = 0.14 nM T02551 CJF9H4 25186569 Ki = 0.099 nM T02551 CG6NC3 25186839 Ki = 32.92 nM T02551 C78HME 25212275 Ki = 15 nM T02551 CE6Z9I 25212276 Ki = 149 nM T02551 COV83Z 25256814 Ki = 1.7 nM T02551 C76ROY 25256815 Ki = 6.761 nM T02551 C7JZ2D 25256816 Ki = 0.27 nM T02551 C6PL1Y 25256817 Ki = 14.45 nM T02551 CR89HN 27039365 Ki > 50316 nM T02551 C4MRQ0 27842480 EC50 = 0.18 nM T02551 C60SDV 27846376 EC50 = 22000 nM T02551 C0BJ5F 27846916 EC50 = 9.2 nM T02551 CYG87R 27847327 EC50 = 1000 nM T02551 CDY01I 30982708 Ki = 110 nM T02551 C9R0CK 31281277 EC50 = 2500 nM T02551 C9QGK3 34257212 Ki = 53 nM T02551 CFE27P 35995182 EC50 = 225 nM T02551 C8VRX4 36717024 EC50 = 611 nM T02551 CX8IT3 38417721 EC50 = 155 nM T02551 C20XSK 39729535 EC50 = 550 nM T02551 CY1O0S 41532205 Ki = 67 nM T02551 C0XMS9 42605994 Ki = 19000 nM T02551 CD61JW 42606339 Ki = 8700 nM T02551 C0TN5O 42606573 Ki = 12000 nM T02551 CDE4U8 42609932 Ki = 2.95 nM T02551 C7BPK4 42625205 Ki = 11.3 nM T02551 CS8OZ6 42625207 IC50 = 1.09 nM T02551 CJ2TA7 42625211 IC50 = 6.51 nM T02551 CQ37BN 42625290 Ki = 6.11 nM T02551 CXB28J 42625293 Ki = 7.5 nM T02551 CYM0J6 42625295 Ki = 0.26 nM T02551 CK3QD2 42625354 Ki = 35.8 nM T02551 CD9RN1 42626103 Ki = 0.44 nM T02551 CTW8G4 42626171 Ki = 5.21 nM T02551 C0P3JR 42626172 Ki = 0.92 nM T02551 CZ19KX 42626240 Ki = 3.9 nM T02551 CTL2I7 42626243 Ki = 1.61 nM T02551 CLH7Y0 42626289 Ki = 30 nM T02551 C5VTZ6 42626293 Ki = 80 nM T02551 C98BKP 42626313 Ki = 7.51 nM T02551 C1VR4S 42626315 Ki = 4.6 nM T02551 CRMZ20 42626317 Ki = 0.51 nM T02551 CRQ91B 42626318 Ki = 0.53 nM T02551 CTYZ17 42626380 Ki = 3.6 nM T02551 C1JK6E 42626381 IC50 = 1.58 nM T02551 C0AI7N 43229249 Ki = 161 nM T02551 C75LHU 43398192 Ki > 50000 nM T02551 CEL6J0 44123782 Ki = 11 nM T02551 C2AV1K 44190762 IC50 = 837 nM T02551 C6SG0O 44192200 Ki = 1316 nM T02551 CS4TB9 44203057 Ki = 6.3 nM T02551 CMR7T1 44204999 Ki = 1.259 nM T02551 CVG6X1 44209472 Ki = 229 nM T02551 CD5AB7 44209480 Ki = 86 nM T02551 CBA7V5 44212307 Ki = 1.995 nM T02551 CM76LY 44212310 Ki = 0.7943 nM T02551 CJ50AI 44212312 Ki = 5.012 nM T02551 COS94W 44222483 Ki = 3.4 nM T02551 CNW3R8 44222488 Ki = 220 nM T02551 C1ST2I 44241718 Ki = 310 nM T02551 CJ8RW5 44249745 Ki = 0.7943 nM T02551 C2FDB1 44250364 IC50 > 10000 nM T02551 C8MC0Q 44251387 IC50 > 10000 nM T02551 C5YEA8 44251388 IC50 > 10000 nM T02551 C0BSF6 44251389 IC50 > 10000 nM T02551 C2K0VZ 44253016 Ki > 501.19 nM T02551 C1C0JQ 44263882 Ki = 5200 nM T02551 CQ13GA 44264622 Ki = 6600 nM T02551 CMP0F2 44264623 Ki = 5300 nM T02551 CHGO69 44264629 Ki = 21000 nM T02551 CKD0E4 44264641 Ki = 34000 nM T02551 C41LTK 44264642 Ki = 230 nM T02551 CJI76B 44264644 Ki = 1100 nM T02551 CS4YW5 44264682 Ki = 560 nM T02551 CCK6Z0 44264741 Ki = 61000 nM T02551 C6LNX8 44264742 Ki = 5500 nM T02551 C43LUM 44270444 Ki = 9400 nM T02551 CWK09J 44270558 Ki = 3715.35 nM T02551 CK7A9H 44274130 Ki = 19.95 nM T02551 CSIM26 44274174 Ki = 19.95 nM T02551 CQD08W 44274186 Ki = 794.33 nM T02551 CMI4G9 44275820 Ki = 292 nM T02551 CFP7Z8 44276050 Ki = 9 nM T02551 CE10KM 44276075 Ki = 4.7 nM T02551 CTM39J 44276079 Ki = 20 nM T02551 CQ8V6N 44276105 Ki = 163 nM T02551 C3AS0H 44276111 Ki = 19 nM T02551 CK2R3A 44276536 Ki = 0.9 nM T02551 C0JPB1 44277402 Ki = 652 nM T02551 CSB0G2 44277403 Ki = 24 nM T02551 CN1X3R 44277404 Ki = 731 nM T02551 CX9PO7 44277421 Ki = 652 nM T02551 CGD2I6 44277524 Ki = 251.19 nM T02551 CQV0T7 44277529 Ki = 50.12 nM T02551 CXLV91 44277535 Ki = 316.23 nM T02551 C27ULI 44277569 Ki > 10000 nM T02551 CF28KD 44277580 Ki = 270 nM T02551 C4RG7F 44277587 Ki > 10000 nM T02551 C4HWK2 44277588 Ki = 251.19 nM T02551 CGY34K 44277819 Ki = 731 nM T02551 C84TMG 44278427 Ki = 457 nM T02551 CI37UT 44278788 Ki = 537 nM T02551 C8Q5RI 44283757 Ki > 3000 nM T02551 C1T2BY 44283889 Ki > 3000 nM T02551 CZF8B5 44283891 Ki > 3000 nM T02551 C5WHP1 44283941 Ki > 3000 nM T02551 CK5TX4 44297323 Ki = 3.162 nM T02551 C5NK9B 44297390 Ki = 5.012 nM T02551 CSKN61 44297458 Ki = 25.12 nM T02551 CZR0L7 44297472 Ki = 39.81 nM T02551 C4G8QT 44297494 Ki = 10 nM T02551 CL5H8S 44297514 Ki = 2.512 nM T02551 CTK86W 44297596 Ki = 50.12 nM T02551 CJD36K 44297665 Ki = 125.89 nM T02551 C5U0KI 44297693 Ki = 2.512 nM T02551 CWNI02 44297694 Ki = 1.995 nM T02551 C5X1PJ 44297720 Ki = 50.12 nM T02551 CBSQ04 44300865 Ki = 514 nM T02551 CQ5A2E 44301054 Ki = 1800 nM T02551 CNW2F3 44304314 IC50 = 4000 nM T02551 CWJA31 44304603 Ki = 115 nM T02551 CK8QJ6 44304621 Ki = 120 nM T02551 CR9SB5 44304643 Ki = 1200 nM T02551 CH6FM8 44304644 Ki = 1300 nM T02551 CGY80N 44304652 Ki = 660 nM T02551 CKBE16 44304814 Ki = 5850 nM T02551 C61YBG 44305039 Ki = 7.943 nM T02551 CIC7S0 44305123 Ki = 19.95 nM T02551 CHEO59 44305138 Ki = 25.12 nM T02551 C1V7ER 44305156 Ki = 6.31 nM T02551 C2XMP1 44305196 Ki = 6.31 nM T02551 CKX85J 44305348 Ki = 0.7943 nM T02551 CU7J1E 44305390 Ki = 0.631 nM T02551 CGP8X5 44309509 Ki = 1.4 nM T02551 CM92JC 44309510 Ki = 1.6 nM T02551 CP1QG5 44309688 Ki = 8.2 nM T02551 CKY68S 44309775 Ki = 1.5 nM T02551 C1TKV6 44309876 Ki = 0.28 nM T02551 CRD9Z2 44310792 Ki = 6.31 nM T02551 C9GLP3 44311009 Ki = 3.162 nM T02551 C6RF1P 44316315 Ki = 16 nM T02551 CL6KC8 44317000 Ki = 22 nM T02551 CRIT59 44317001 Ki = 24 nM T02551 C47HKR 44317002 Ki = 32 nM T02551 C60LKZ 44317003 Ki = 19.7 nM T02551 CL3B1F 44317030 Ki = 4.3 nM T02551 C2J1GU 44317031 Ki = 2.4 nM T02551 C9LF3J 44317054 Ki = 2 nM T02551 C2XY0L 44317069 Ki = 3.2 nM T02551 C1HK5Z 44317088 Ki = 8 nM T02551 C1VLM3 44317105 Ki = 0.5 nM T02551 CG9FT0 44317222 Ki = 85 nM T02551 C6JMU9 44317229 Ki = 4.2 nM T02551 CA2ZM7 44317252 Ki = 6 nM T02551 CXK60V 44317260 Ki = 15 nM T02551 C3CZD1 44317272 Ki = 4.7 nM T02551 C9ZK2O 44317275 Ki = 5 nM T02551 C6TC3I 44317294 Ki = 4.7 nM T02551 C9DKH3 44317295 Ki = 5.2 nM T02551 CVP35Q 44317384 Ki = 1.4 nM T02551 CO6I2J 44317385 Ki = 0.6 nM T02551 CZ6O2I 44317425 Ki = 2.5 nM T02551 CDI5G8 44317436 Ki = 4.8 nM T02551 CT7S5Y 44317450 Ki = 4 nM T02551 CBW78P 44317467 Ki = 1.4 nM T02551 CTFO42 44317468 Ki = 12.4 nM T02551 CV8WZ0 44318454 IC50 = 14.13 nM T02551 CXJL56 44318842 IC50 > 1000 nM T02551 CWUE26 44319102 Ki = 690 nM T02551 CTE14R 44319217 Ki = 18 nM T02551 C8LXY4 44319269 Ki = 87 nM T02551 CV2UN7 44319361 Ki = 1200 nM T02551 CN1M5O 44319362 Ki = 1201 nM T02551 CC2W9S 44319368 Ki = 1000 nM T02551 CCD3V1 44319369 Ki = 710 nM T02551 CY9ZX7 44319370 Ki = 2500 nM T02551 CUB9J4 44319412 Ki = 2000 nM T02551 C3Z9BT 44319418 Ki = 275 nM T02551 C82GVM 44319482 Ki > 2040 nM T02551 CC2GZ0 44319568 Ki = 19 nM T02551 C31IGQ 44319569 Ki = 131 nM T02551 CJ02KH 44319612 Ki = 39 nM T02551 CK0D6E 44319723 Ki = 3.981 nM T02551 CU06KP 44319980 Ki = 15.85 nM T02551 C5YA0V 44321001 Ki > 8000 nM T02551 CG5E2U 44323763 Ki = 14.7 nM T02551 CY1I0M 44323780 Ki = 591.3 nM T02551 CW16JD 44324737 Ki = 107 nM T02551 CA84SN 44324765 Ki = 270 nM T02551 COA3H4 44324800 Ki = 433 nM T02551 CLDK96 44324801 Ki = 125.89 nM T02551 C2SMT6 44324802 Ki = 12.59 nM T02551 CY04JW 44324972 Ki = 611 nM T02551 C3UWI1 44324978 Ki = 10 nM T02551 C0Z1NV 44324979 Ki = 7.943 nM T02551 CCT67J 44324980 Ki = 1.1 nM T02551 CB5H2S 44324986 Ki = 3.162 nM T02551 CUZ67X 44325021 Ki = 25.12 nM T02551 CN07UQ 44325025 Ki = 0.7943 nM T02551 CI30DU 44325026 Ki = 15.85 nM T02551 C8KWG4 44325037 Ki = 15.85 nM T02551 CGL51N 44325577 Ki = 67 nM T02551 CXPS18 44325578 Ki = 61 nM T02551 COM07T 44325658 Ki = 22 nM T02551 CQE81D 44325894 Ki > 455 nM T02551 CE0S1Z 44325900 Ki > 1500 nM T02551 CKW98Z 44325908 Ki = 56 nM T02551 CV56DM 44326256 Ki = 27 nM T02551 CV8A2N 44326257 Ki = 45 nM T02551 C2X9GN 44326324 Ki = 323 nM T02551 CHVF93 44329039 Ki = 770 nM T02551 C1Y4VO 44329046 Ki = 199.53 nM T02551 C69IHO 44329050 Ki = 251.19 nM T02551 CFA61T 44329053 Ki = 15.85 nM T02551 C75IBH 44329057 Ki = 676.08 nM T02551 CZX74M 44329058 Ki = 251.19 nM T02551 CT8KH0 44329062 Ki = 794.33 nM T02551 C8NA9T 44329067 Ki = 501.19 nM T02551 C5NOQ0 44329068 Ki = 15.85 nM T02551 CB8J3N 44329090 Ki = 1800 nM T02551 C6G3SV 44329093 Ki = 323.59 nM T02551 CF0AN3 44329097 Ki = 1400 nM T02551 CXQK21 44329098 Ki = 8511.38 nM T02551 C6MP1F 44329099 Ki = 1445.44 nM T02551 CM9NS0 44329102 Ki = 50.12 nM T02551 CI2Z9F 44329106 Ki = 6.31 nM T02551 COL9X4 44329121 Ki = 1258.93 nM T02551 C5QOA8 44329126 Ki = 50.12 nM T02551 CT7CZ6 44329130 Ki = 12.59 nM T02551 CR5FP1 44329136 Ki = 630.96 nM T02551 C50WAC 44329282 Ki = 590 nM T02551 CF3C7Y 44329283 Ki = 416.87 nM T02551 C7WOC9 44329284 Ki = 3600 nM T02551 CGOY38 44329293 Ki = 912.01 nM T02551 CE62MT 44329299 Ki = 724.44 nM T02551 CK7WF9 44329312 Ki = 9700 nM T02551 CM52IE 44329314 Ki = 416.87 nM T02551 C1WYS3 44329321 Ki = 1 nM T02551 C90PLN 44329483 Ki = 29 nM T02551 C5J3PW 44329749 Ki = 1.56 nM T02551 C6NH5U 44329754 Ki > 10000 nM T02551 C6H4BO 44332565 Ki = 11 nM T02551 C9JQK3 44332566 Ki > 1000 nM T02551 C1E7KI 44332581 Ki = 281.5 nM T02551 CD7N6W 44332613 Ki > 400 nM T02551 COR0D5 44332646 Ki > 5000 nM T02551 C63TDB 44332686 Ki = 42.5 nM T02551 COG5D1 44332701 Ki = 27.8 nM T02551 CZ6F4T 44333001 Ki = 12 nM T02551 C0UT6E 44333374 Ki = 240 nM T02551 C9MVH8 44333746 Ki = 3000 nM T02551 CFT4L1 44336552 Ki = 5100 nM T02551 CS3TZ4 44336571 Ki = 7000 nM T02551 CD42FX 44337659 Ki > 8000 nM T02551 CT3M2R 44337675 Ki = 4010 nM T02551 CPVO39 44337705 Ki = 6100 nM T02551 C2ECI8 44337709 Ki = 2520 nM T02551 C5S9WU 44337725 Ki = 193 nM T02551 C0ZH4Y 44338149 Ki = 214 nM T02551 CQ0ZF9 44338248 Ki = 53.2 nM T02551 C1I8XF 44339879 Ki = 560 nM T02551 C34CBZ 44339953 Ki = 20 nM T02551 CPF62D 44339984 Ki = 140 nM T02551 CIS79K 44339992 Ki = 130 nM T02551 C84OZX 44340084 Ki = 13 nM T02551 C9I7GN 44340097 Ki = 27 nM T02551 CBQ3D5 44340186 Ki = 2900 nM T02551 CT5HC3 44340227 Ki = 33 nM T02551 C7-SEP 44340278 Ki = 10 nM T02551 C1EZY8 44340285 Ki = 3.162 nM T02551 C6LDF1 44340301 Ki = 31.62 nM T02551 C5HGU2 44340302 Ki = 580 nM T02551 CA71HQ 44340333 Ki = 79 nM T02551 CJL8H0 44340337 Ki = 10 nM T02551 C8RN4J 44340352 Ki = 1.585 nM T02551 CFRK78 44340353 Ki = 10 nM T02551 CUG2V9 44340354 Ki = 2.512 nM T02551 CA1F3K 44340364 Ki = 6.31 nM T02551 CQPW26 44340376 Ki = 410 nM T02551 C3QW1F 44340415 Ki = 1000 nM T02551 CO2QV3 44340654 Ki = 1.585 nM T02551 CLK24X 44340661 Ki = 50.12 nM T02551 C8FC4J 44340690 Ki = 2.512 nM T02551 C2N0UR 44340694 Ki = 100 nM T02551 CPOL72 44340695 Ki = 0.631 nM T02551 CS48JN 44340705 Ki = 12.59 nM T02551 C8QYA4 44340965 Ki = 0.1995 nM T02551 CC2D6N 44340967 Ki = 0.3981 nM T02551 CB2G0T 44340985 Ki = 7.943 nM T02551 CD9ZS8 44342270 IC50 = 154 nM T02551 C6N3XK 44345317 IC50 < 1000 nM T02551 C5GW8X 44350679 Ki = 38 nM T02551 CTXY90 44350788 Ki = 0.5 nM T02551 CZX4S1 44350839 Ki = 6.6 nM T02551 C4QP5U 44350942 Ki = 125 nM T02551 C50HVX 44350991 Ki = 374 nM T02551 CUGT13 44351005 Ki = 1.48 nM T02551 C8SX6R 44353325 Ki = 5.012 nM T02551 C0ZYJ5 44353345 Ki = 3.981 nM T02551 C9S7RU 44353346 Ki = 501.19 nM T02551 CFIO91 44353352 Ki = 1 nM T02551 C65MOI 44353353 Ki = 3.162 nM T02551 C06VLC 44353354 Ki = 10 nM T02551 CAF53W 44353361 Ki = 25.12 nM T02551 CI2HW1 44353363 Ki = 3.981 nM T02551 CH94PY 44353393 Ki = 7.943 nM T02551 C4DEX7 44353394 Ki = 630.96 nM T02551 CO6J8B 44353397 Ki = 3162.28 nM T02551 CGA62E 44353398 Ki = 12.59 nM T02551 CX02GJ 44353399 Ki = 25.12 nM T02551 CVK1R7 44353406 Ki = 6.31 nM T02551 C76VOZ 44353407 Ki = 1584.89 nM T02551 CR7V1I 44353412 Ki = 1.995 nM T02551 CWQ51L 44353425 Ki = 50.12 nM T02551 CM1Y8U 44353431 Ki = 6.31 nM T02551 CAQC14 44353432 Ki = 6.31 nM T02551 CULV76 44353438 Ki = 63.1 nM T02551 CJ95DV 44353440 Ki = 19.95 nM T02551 CWX5J3 44353475 Ki = 3.162 nM T02551 CJ0AS5 44353476 Ki = 3.981 nM T02551 CEOI46 44353477 Ki = 1.995 nM T02551 C5FQP1 44353479 Ki = 19.95 nM T02551 CDK4M0 44353487 Ki = 0.1585 nM T02551 CU67QT 44353488 Ki = 1.259 nM T02551 CZV3S0 44355355 Ki = 154 nM T02551 CNV5M9 44355433 Ki = 211 nM T02551 C9W5AB 44356064 Ki = 113 nM T02551 CP38IC 44356249 Ki = 30.2 nM T02551 C9GB5E 44356253 Ki = 0.5 nM T02551 CS7P5O 44357894 Ki = 1.1 nM T02551 CJ80OW 44360984 Ki = 19.95 nM T02551 CS8K1A 44360992 Ki = 28.84 nM T02551 C3NZ7B 44361021 Ki = 2.8 nM T02551 CL2RI0 44363213 Ki = 1.995 nM T02551 C8WJ7M 44363215 Ki = 6.31 nM T02551 CIS8Z4 44363218 Ki = 39.81 nM T02551 COY57L 44363232 Ki = 6.31 nM T02551 CTM6J0 44363348 Ki = 3.981 nM T02551 C9ZB4M 44370009 Ki = 1100 nM T02551 C81CTM 44370032 Ki = 25 nM T02551 C50OBQ 44370047 Ki = 50 nM T02551 C4JCY7 44370058 Ki = 530 nM T02551 C0DQS7 44371025 Ki = 50.2 nM T02551 CU49IQ 44371356 Ki = 55.7 nM T02551 CR5IM4 44371566 Ki = 756 nM T02551 C6PSR0 44371932 Ki = 5900 nM T02551 CQ1IU6 44371980 Ki = 270 nM T02551 C2JFZ9 44371996 Ki = 410 nM T02551 CK6GM7 44371997 Ki = 17000 nM T02551 CXZ6A7 44372009 Ki = 840 nM T02551 C4VLE2 44372153 Ki = 3100 nM T02551 CJXL12 44372154 Ki = 3800 nM T02551 C4O3LX 44372198 Ki = 5700 nM T02551 CZV9O7 44372296 Ki = 2570.4 nM T02551 C1SWI7 44372312 Ki > 100000 nM T02551 CX2B6A 44372338 Ki = 2000 nM T02551 C3GJM6 44374188 Ki = 25.12 nM T02551 C39OSY 44374408 Ki = 63.1 nM T02551 C6L9AR 44374409 Ki = 10 nM T02551 C20MKC 44374410 Ki = 7.943 nM T02551 CAJ92G 44374411 Ki = 3.162 nM T02551 CD5E1G 44374431 Ki = 253 nM T02551 CK28HY 44374637 Ki = 40 nM T02551 C8EK9X 44374648 Ki = 171 nM T02551 C8QLR2 44380405 Ki = 79.43 nM T02551 C8K6BV 44380433 Ki = 251.19 nM T02551 C6X7HM 44380644 Ki = 39.81 nM T02551 CBS4E9 44380645 Ki = 199.53 nM T02551 CF1O8S 44380675 Ki = 125.89 nM T02551 CYI39O 44380685 Ki = 2200 nM T02551 CTY0L5 44380687 Ki = 199.53 nM T02551 CL1ER5 44380697 Ki = 570 nM T02551 C6B9PA 44380715 Ki = 47 nM T02551 CNSG64 44380716 Ki = 11000 nM T02551 C6MWD2 44380717 Ki = 2700 nM T02551 C2FQB1 44380739 Ki = 50.12 nM T02551 C4JGZ2 44380747 Ki = 251.19 nM T02551 CA5EW9 44380770 Ki = 31 nM T02551 C68MUE 44380774 Ki = 210 nM T02551 C4DGR5 44380785 Ki = 570 nM T02551 CUV90Q 44380802 Ki = 320 nM T02551 CCL54M 44380815 Ki = 110 nM T02551 CM01SN 44380816 Ki = 1100 nM T02551 CBHE80 44380836 Ki = 501.19 nM T02551 CLUP31 44380906 Ki = 1000 nM T02551 CT02DY 44380921 Ki = 350 nM T02551 C7KQ3H 44380934 Ki = 1584.89 nM T02551 CAV5J3 44380938 Ki = 398.11 nM T02551 CK3F4H 44381103 Ki = 19.95 nM T02551 C6PI1L 44381117 Ki = 8700 nM T02551 CJ6I0B 44381118 Ki = 360 nM T02551 CN9E8B 44381120 Ki = 100 nM T02551 C6QI1Y 44381124 Ki = 316.23 nM T02551 CBYQ74 44381146 Ki = 7200 nM T02551 C8GA2E 44381147 Ki = 270 nM T02551 C6SDO5 44381216 Ki = 13000 nM T02551 C4OAD2 44381217 Ki = 7400 nM T02551 C67SRD 44381276 Ki = 20000 nM T02551 CKR9B8 44381279 Ki = 12000 nM T02551 COB6T7 44381286 Ki = 1900 nM T02551 CZ7Q2X 44381424 Ki = 12000 nM T02551 CQO5G1 44381432 Ki = 3300 nM T02551 CI0YA1 44382105 Ki < 10000 nM T02551 CPDA94 44382118 Ki = 125.89 nM T02551 CRK0U1 44382163 Ki = 199.53 nM T02551 CF7E9O 44382164 Ki = 79.43 nM T02551 C5CG2L 44382165 Ki = 63.1 nM T02551 CSC5Z4 44382774 Ki < 10000 nM T02551 C7KW3P 44382826 Ki < 10000 nM T02551 CUL1Y2 44382827 Ki < 10000 nM T02551 C5H4KM 44382828 Ki = 25.12 nM T02551 C8L5WN 44382829 Ki = 501.19 nM T02551 CQ85AW 44389003 Ki = 627 nM T02551 C8AG7U 44389016 Ki = 741 nM T02551 CEO2W9 44393372 Ki = 0.86 nM T02551 CXP4Q7 44393393 Ki = 1.4 nM T02551 C6BZS0 44393403 Ki = 0.72 nM T02551 C86NED 44393411 Ki = 4.5 nM T02551 C9THO4 44393415 Ki = 2.4 nM T02551 C8EC7R 44395709 Ki > 10000 nM T02551 CF7I1C 44395711 Ki = 172 nM T02551 C3RV6T 44395741 Ki = 180 nM T02551 C4B0OI 44397588 Ki = 1000 nM T02551 C5FP0R 44397589 Ki = 1584.89 nM T02551 CE3G8U 44397670 Ki = 630.96 nM T02551 CBD9Z1 44399901 Ki = 43.65 nM T02551 CFYO16 44399902 Ki = 38.9 nM T02551 C0E5HY 44400500 Ki = 2 nM T02551 CO8EU5 44400519 Ki = 0.84 nM T02551 CRX12E 44400553 Ki = 3.5 nM T02551 CIU18E 44400585 EC50 = 3.9 nM T02551 CV8K2W 44400594 Ki = 20 nM T02551 C84RNU 44400626 EC50 = 3.5 nM T02551 CY94SF 44400674 EC50 = 2 nM T02551 CX7O9S 44401041 Ki = 31 nM T02551 C5XC2B 44401042 Ki = 45 nM T02551 CD56EA 44401105 Ki = 95 nM T02551 CW3PC2 44401106 Ki = 8.6 nM T02551 C9WH7P 44401164 Ki = 1.1 nM T02551 C9CWX1 44401194 Ki = 293 nM T02551 CXT84G 44401243 Ki = 251 nM T02551 C1B4QL 44403095 Ki > 10000 nM T02551 C1YL7Z 44403098 Ki > 10000 nM T02551 CFV98A 44403101 Ki > 10000 nM T02551 C6OY9S 44403102 Ki > 10000 nM T02551 CH4SX6 44403105 Ki > 10000 nM T02551 C12FIH 44403106 Ki > 10000 nM T02551 CQ4U2P 44403210 Ki = 4.3 nM T02551 CKE6T4 44403213 Ki = 0.53 nM T02551 CAJX39 44403214 Ki = 14 nM T02551 C61CNS 44403219 Ki = 1.1 nM T02551 C5AE9L 44403220 Ki = 86 nM T02551 CC6XM4 44403224 Ki = 9 nM T02551 C6JB4M 44403225 Ki = 210 nM T02551 CGE52H 44403232 Ki = 16 nM T02551 C4LKC1 44404394 Ki > 10000 nM T02551 C3EJ4G 44404396 Ki > 10000 nM T02551 CRQ1J7 44406885 Ki = 4.4 nM T02551 COL64Y 44406886 Ki = 3.4 nM T02551 CSJ95I 44406895 Ki = 2.3 nM T02551 C0NHR2 44406899 Ki = 5.4 nM T02551 CT57XV 44406913 Ki = 1.7 nM T02551 CV8YF1 44406926 Ki = 4.8 nM T02551 CVU15M 44406983 Ki = 3.7 nM T02551 CPE1L4 44406984 Ki = 7.4 nM T02551 CH8L2V 44407007 Ki = 7.4 nM T02551 C8WD1P 44407270 Ki = 3.4 nM T02551 CDG04R 44407298 Ki = 58.9 nM T02551 C16HAY 44407300 Ki = 64.9 nM T02551 CVK80E 44407307 Ki = 22.4 nM T02551 C5HYM0 44407308 Ki = 12.1 nM T02551 C4WM7J 44407319 Ki = 4054 nM T02551 C8VHO1 44407320 Ki = 9.2 nM T02551 C8QXI0 44407346 Ki = 4.5 nM T02551 CN52HW 44407347 Ki = 3.9 nM T02551 CCS63V 44407363 Ki = 2.5 nM T02551 C3V5TA 44407424 Ki = 10.1 nM T02551 C8SA0E 44407425 Ki = 11.2 nM T02551 CA64GU 44407436 Ki = 16.8 nM T02551 C74XRS 44407437 Ki = 9.6 nM T02551 CAX81F 44407442 Ki = 293 nM T02551 CZ24HP 44408818 Ki = 75.7 nM T02551 C7AC1M 44409606 Ki = 11.4 nM T02551 C12HNJ 44409613 Ki = 2.7 nM T02551 C5A8GN 44409704 Ki = 9.3 nM T02551 CV9HI5 44409706 Ki = 8.3 nM T02551 C1AMJ7 44409707 Ki = 6.2 nM T02551 C9HR5I 44409720 Ki = 7.9 nM T02551 CR7XG9 44409721 Ki = 2.2 nM T02551 CDXJ02 44409726 Ki = 2.3 nM T02551 CKMT45 44409727 Ki = 7.2 nM T02551 CJ6LU7 44409730 Ki = 6.7 nM T02551 C4G9ZY 44409731 Ki = 0.9 nM T02551 CDW31B 44409888 Ki = 12.1 nM T02551 C31CNO 44409890 Ki = 4 nM T02551 C8V2XC 44409891 Ki = 5.5 nM T02551 CL26QH 44409908 Ki = 1.6 nM T02551 CP81TR 44409911 Ki = 3.2 nM T02551 C0VZ1B 44409913 Ki = 35.7 nM T02551 CJD14X 44409925 Ki = 32.2 nM T02551 CR2CJ9 44412182 Ki = 360 nM T02551 CF9IW1 44412191 Ki = 320 nM T02551 C8FU9P 44412268 Ki = 1200 nM T02551 C78RSG 44412269 Ki = 340 nM T02551 CKY57Q 44412458 Ki = 94 nM T02551 CK9FC8 44412468 Ki = 158.49 nM T02551 C63XKI 44412482 Ki = 72 nM T02551 C2UBR0 44412494 Ki = 1900 nM T02551 CCPO37 44419053 Ki = 0.389 nM T02551 CGL9E1 44419056 Ki = 0.3802 nM T02551 CP5M3H 44419060 Ki = 4.266 nM T02551 CJ4EZ9 44419065 Ki = 33.11 nM T02551 CIWX27 44419066 Ki = 93.33 nM T02551 CE2V0S 44425698 Ki = 39.81 nM T02551 C2TE3S 44425699 Ki = 19.95 nM T02551 C90AOQ 44425700 Ki = 25.12 nM T02551 CU52GB 44425701 Ki = 1.995 nM T02551 C9F1XP 44425702 Ki = 3.981 nM T02551 CR1QN5 44425703 Ki = 15.85 nM T02551 C5UZS7 44425704 Ki = 25.12 nM T02551 CN96FA 44425705 Ki = 15.85 nM T02551 C1J9MY 44425706 Ki = 1.585 nM T02551 CPI52U 44425708 Ki = 3.981 nM T02551 CNZ3M7 44425711 Ki = 5.012 nM T02551 C92AZG 44425714 Ki = 2.512 nM T02551 C7LP1B 44425717 Ki = 0.7943 nM T02551 CX8TR0 44425719 Ki = 3.162 nM T02551 CJN6P4 44427818 Ki = 0.4 nM T02551 CW3F5H 44427820 Ki = 0.6 nM T02551 CYLO03 44427821 Ki = 1.4 nM T02551 CJY9L5 44427822 Ki = 1.6 nM T02551 CO46HS 44427823 Ki = 1.1 nM T02551 CFG0S3 44427824 Ki = 49.2 nM T02551 C7PK0M 44427825 Ki = 2.9 nM T02551 CDV6A3 44427826 Ki = 1.2 nM T02551 C65ZXC 44427827 EC50 = 1 nM T02551 CZ0X7U 44427829 Ki = 1.8 nM T02551 C9U8YT 44427831 Ki = 2.8 nM T02551 C0C8AH 44427835 EC50 = 3.9 nM T02551 C8EV3G 44427836 Ki = 0.5 nM T02551 CA96WP 44427839 Ki = 2.5 nM T02551 C46BRT 44427840 Ki = 1.3 nM T02551 CS9ND5 44427841 Ki = 1 nM T02551 COV6N3 44427842 Ki = 160 nM T02551 CY0QJ2 44427970 Ki = 14830 nM T02551 CCRH08 44428207 Ki = 1.585 nM T02551 C2AZ6B 44436300 Ki = 66 nM T02551 C30QMX 44436301 Ki = 287 nM T02551 C9AJ0D 44436302 Ki = 187 nM T02551 C3NVL0 44436303 Ki = 527 nM T02551 CREM27 44436304 Ki = 1780 nM T02551 C53XYK 44436305 Ki = 102 nM T02551 C2LF9K 44436306 Ki = 247 nM T02551 C9H8ST 44436307 Ki = 660 nM T02551 C7IBE2 44436308 Ki = 14 nM T02551 C2B4WN 44436596 Ki = 31 nM T02551 CLV2E1 44436597 Ki = 29 nM T02551 C0LBO6 44436598 Ki = 50 nM T02551 CREV94 44436599 Ki = 68 nM T02551 CZ37MU 44436600 Ki = 1 nM T02551 CRW39P 44436601 Ki = 10 nM T02551 CG06FU 44436602 Ki = 6.2 nM T02551 C2GD0Z 44436603 Ki = 22 nM T02551 C1T9IF 44436605 Ki = 0.31 nM T02551 CBQ6F7 44436606 Ki = 3.2 nM T02551 C6ZJ1W 44436608 Ki = 0.83 nM T02551 C1OP6H 44436610 Ki = 7.5 nM T02551 CR6UK2 44436617 Ki = 37 nM T02551 CHTG80 44436618 Ki = 1.5 nM T02551 CI5K6A 44436621 Ki = 5.6 nM T02551 CW7VF4 44436719 Ki = 133 nM T02551 CP85SY 44436720 Ki = 42.9 nM T02551 C1J6BZ 44436721 Ki = 11.1 nM T02551 C8I7HR 44436722 Ki = 30.3 nM T02551 CLU0F7 44436723 Ki = 28.4 nM T02551 CE0M4N 44436724 Ki = 30.2 nM T02551 CR7Y8E 44436725 Ki = 2.82 nM T02551 CFP41N 44436726 Ki = 2.4 nM T02551 C7QH5X 44436727 Ki = 17.7 nM T02551 C04VDB 44436728 Ki = 38.9 nM T02551 C4ZN9T 44436729 Ki = 12.3 nM T02551 C2V4IE 44436730 Ki = 32.6 nM T02551 C4ZN9E 44436731 Ki = 40.9 nM T02551 C29BYE 44436732 Ki = 36.9 nM T02551 C6UWG1 44436735 Ki = 340 nM T02551 C4GX5V 44436737 Ki = 3.6 nM T02551 C9YC8V 44436739 Ki = 15.2 nM T02551 CDT72W 44436741 Ki = 15.2 nM T02551 C1J2MR 44436743 Ki = 22.8 nM T02551 C4HR8W 44436745 Ki > 1000 nM T02551 CZ6H2Q 44436746 Ki = 50.2 nM T02551 CAD4I1 44436747 Ki > 1000 nM T02551 C8PX3T 44436748 Ki = 500 nM T02551 C8BO7G 44436750 Ki > 1000 nM T02551 C5L3JM 44436751 Ki = 99.1 nM T02551 CXI70P 44436753 Ki = 10.9 nM T02551 CGP8C7 44436756 Ki = 6.01 nM T02551 C6K9DT 44436759 Ki = 2.7 nM T02551 CCL5K1 44436762 Ki > 1000 nM T02551 CZ5V0R 44436765 Ki = 31.1 nM T02551 C7Y5VG 44436767 Ki = 2340 nM T02551 CN49HQ 44436768 Ki > 1000 nM T02551 C06RTZ 44436769 Ki > 1000 nM T02551 C6JQ1H 44436771 Ki = 18.4 nM T02551 CN2Q5J 44436772 Ki = 10.8 nM T02551 CG2X1D 44437896 Ki = 11 nM T02551 CX04CK 44437897 Ki = 22 nM T02551 CC4V7G 44438186 Ki = 1860 nM T02551 CJ8W5C 44438197 EC50 = 232 nM T02551 CMGT04 44438199 Ki = 450 nM T02551 C8C0HP 44438201 EC50 = 41.5 nM T02551 CJDT47 44438203 Ki = 570 nM T02551 CU4AS8 44438204 Ki = 490 nM T02551 CPAE72 44438206 Ki = 16800 nM T02551 CJM3K5 44438208 Ki = 2130 nM T02551 CPH7V5 44438209 Ki = 1950 nM T02551 C6K3ZU 44438210 Ki = 467 nM T02551 CADG24 44438211 Ki = 2100 nM T02551 CLE5G1 44438213 Ki = 5480 nM T02551 C8ILG5 44438215 Ki = 4270 nM T02551 CFE50G 44438218 EC50 = 347 nM T02551 C3KS0B 44438219 Ki = 382 nM T02551 CAQ5Y9 44438220 Ki = 193 nM T02551 C52KTZ 44438221 Ki = 211 nM T02551 C8LW2C 44438222 Ki = 684 nM T02551 CF2WK6 44438223 Ki = 544 nM T02551 CVT06Y 44438224 Ki = 724 nM T02551 C4POI0 44438225 Ki > 5000 nM T02551 CO76KJ 44438226 Ki = 12500 nM T02551 CJZ69F 44438227 Ki = 106 nM T02551 CS1H8X 44438228 EC50 = 248 nM T02551 CEQ1L8 44438229 Ki = 718 nM T02551 CUF21H 44438230 EC50 = 20.2 nM T02551 CU49FT 44438231 Ki = 156 nM T02551 CD89OH 44438232 Ki = 440 nM T02551 C0VA9W 44438233 Ki = 28 nM T02551 CJSX04 44438234 Ki = 53 nM T02551 CWE9K4 44438235 Ki = 139 nM T02551 C5Q6PG 44438236 EC50 = 98.6 nM T02551 CWS8R5 44438237 Ki = 488 nM T02551 CL4FV8 44438239 Ki = 638 nM T02551 CKZF16 44439165 Ki = 1995.26 nM T02551 CA4HZ3 44439167 Ki = 1258.93 nM T02551 CBI86V 44439942 Ki = 475 nM T02551 C3HMI2 44439943 Ki = 944 nM T02551 C63PQV 44439944 Ki = 1135 nM T02551 C2P4CI 44439945 Ki = 2070 nM T02551 C1UAM5 44443901 EC50 = 864 nM T02551 CU96SV 44443902 EC50 = 547 nM T02551 CIJ85M 44443903 EC50 = 1312 nM T02551 CZ34PG 44443904 EC50 > 10000 nM T02551 C4BUQ3 44443905 EC50 > 3000 nM T02551 CS21LM 44443907 EC50 > 1000 nM T02551 CQ27IL 44443908 EC50 > 1000 nM T02551 CBL7R2 44443909 EC50 > 1000 nM T02551 C7B6UI 44443910 EC50 > 1000 nM T02551 C8KWH4 44443911 EC50 > 1000 nM T02551 CFWE36 44443912 EC50 > 1000 nM T02551 CG62YW 44443913 EC50 > 1000 nM T02551 CH43IX 44443914 EC50 > 1000 nM T02551 CGM1A8 44443915 EC50 > 1000 nM T02551 CV06CS 44443916 EC50 > 1000 nM T02551 C1TV2U 44443918 EC50 > 1000 nM T02551 CF15SI 44443920 EC50 > 1000 nM T02551 CGPV82 44443922 EC50 > 1000 nM T02551 CTF87I 44443923 EC50 = 35 nM T02551 CXZ80S 44443927 EC50 > 5900 nM T02551 CK0T9J 44443930 EC50 = 37 nM T02551 CEFL05 44443934 EC50 > 10000 nM T02551 CQI0U5 44443940 EC50 > 10000 nM T02551 CDR79T 44443941 EC50 > 10000 nM T02551 C3U2QD 44443942 EC50 > 1000 nM T02551 CKZ6T5 44443943 EC50 > 1000 nM T02551 C5DWN4 44443944 EC50 = 427 nM T02551 C0C8LS 44443945 EC50 > 1000 nM T02551 C84FQM 44443947 EC50 > 1000 nM T02551 CZ4XK0 44443948 EC50 = 40 nM T02551 CSOP82 44443950 EC50 > 1000 nM T02551 CA6S4D 44443952 EC50 > 1000 nM T02551 CB1MX2 44454118 Ki = 199.53 nM T02551 CR3IC6 44454120 Ki = 158.49 nM T02551 C5B0IF 44454150 Ki = 316.23 nM T02551 CRD82N 44454166 Ki = 125.89 nM T02551 CMVS90 44454167 Ki = 251.19 nM T02551 C7FY1E 44454168 Ki = 158.49 nM T02551 CW4S3P 44454190 Ki = 1.585 nM T02551 C7H3CL 44454192 Ki = 251.19 nM T02551 CU0N1E 44454217 Ki = 125.89 nM T02551 C9DBA3 44454218 Ki = 316.23 nM T02551 CK01QH 44454219 Ki = 251.19 nM T02551 CLO6X0 44454223 Ki = 158.49 nM T02551 CECR53 44454247 Ki = 316.23 nM T02551 CD4ZU7 44454248 Ki = 199.53 nM T02551 CS2N1D 44454275 Ki = 316.23 nM T02551 CJ5XB1 44454278 Ki = 2511.89 nM T02551 C4GON0 44454309 Ki = 251.19 nM T02551 C91PHS 44454318 Ki = 398.11 nM T02551 CT50UC 44454320 Ki = 158.49 nM T02551 C35WYK 44454339 Ki = 125.89 nM T02551 CZO96M 44454340 Ki > 501.19 nM T02551 C2CIO7 44454351 Ki = 251.19 nM T02551 C9AH1O 44454352 Ki = 199.53 nM T02551 CM8H2G 44454353 Ki < 251.19 nM T02551 C1EZP7 44454358 Ki = 100 nM T02551 CEB84V 44454371 Ki = 125.89 nM T02551 C5EV7Z 44454381 Ki < 251.19 nM T02551 CWC92Y 44454382 Ki < 251.19 nM T02551 CH0S2F 44454384 Ki = 158.49 nM T02551 C32LHE 44454400 Ki = 251.19 nM T02551 CG18KC 44454401 Ki = 39.81 nM T02551 CI0CJ9 44454402 Ki = 316.23 nM T02551 CP34QH 44454403 Ki = 199.53 nM T02551 CW4OX5 44454418 Ki = 6.31 nM T02551 CW1I4Z 44454420 Ki < 125.89 nM T02551 C8TJW4 44454434 Ki = 630.96 nM T02551 CX9U8I 44454443 Ki = 794.33 nM T02551 CXA7W2 44454458 Ki = 12.59 nM T02551 CBGJ08 44454459 Ki > 63.1 nM T02551 CB1P9X 44454685 Ki = 1100 nM T02551 CZJ8G6 44454707 Ki = 1100 nM T02551 CC5SL3 44454709 Ki = 330 nM T02551 CD6M2F 44454710 Ki = 4900 nM T02551 C5V3RI 44454711 Ki = 270 nM T02551 C1GKA2 44454734 Ki = 77 nM T02551 CBD62A 44454735 Ki = 1100 nM T02551 C12XGE 44456400 Ki > 10000 nM T02551 CL1F7V 44459452 Ki = 3000 nM T02551 CF8DR7 44459463 Ki = 450 nM T02551 CQ2IX7 44461606 IC50 > 1000 nM T02551 C9OY3U 44517726 Ki = 2.512 nM T02551 C8C3UM 44533248 Ki = 3.162 nM T02551 C16HEZ 44555445 Ki > 10000 nM T02551 CVA67X 44568347 Ki = 1000 nM T02551 C5SP0Z 44578445 Ki = 600 nM T02551 CVR7A5 44578446 Ki = 220 nM T02551 C5NS6H 44581972 Ki = 812.83 nM T02551 CK8Z1P 44581973 Ki = 776.25 nM T02551 C3UQ9Z 44581974 Ki = 3548.13 nM T02551 CLNB12 44582112 Ki = 489.78 nM T02551 C9I2VT 44582113 Ki = 12.02 nM T02551 CG24ZJ 44582114 Ki = 1513.56 nM T02551 C21GPX 44582115 Ki = 162.18 nM T02551 CQEF30 44582140 Ki = 40.74 nM T02551 C2F1DE 44582177 Ki = 40 nM T02551 CVE23P 44582178 Ki = 398.11 nM T02551 COZ2M5 44582179 Ki = 630.96 nM T02551 CS7P4T 44582187 Ki = 32.36 nM T02551 CH76ID 44582459 Ki = 1584.89 nM T02551 CZMX30 44582460 Ki = 10000 nM T02551 C6A8RM 44582461 Ki = 8317.64 nM T02551 CUGE87 44582462 Ki = 24547.09 nM T02551 C72BQU 44582489 Ki = 2398.83 nM T02551 CEM2D6 44582490 Ki = 208.93 nM T02551 CLHG02 44582491 Ki = 208.93 nM T02551 CN53TE 44582492 Ki = 1096.48 nM T02551 CG50VT 44582493 Ki = 4168.69 nM T02551 C3EJV6 44582516 Ki = 8317.64 nM T02551 C1F6NA 44582517 Ki = 1047.13 nM T02551 CZK49H 44582518 Ki = 389.05 nM T02551 CQ42JI 44582519 Ki = 8912.51 nM T02551 CFW0V8 44589129 Ki > 1000 nM T02551 CCJK60 44589130 Ki = 19.9 nM T02551 C8GY9A 44589131 Ki = 170 nM T02551 CZ8VE0 44589175 Ki = 95.3 nM T02551 C2C7LE 44589176 Ki = 6217 nM T02551 CYF42C 44589177 Ki = 211 nM T02551 C08TSZ 44589178 Ki = 22.1 nM T02551 C6VA9C 44589179 Ki = 47.2 nM T02551 C0LDK7 44589180 Ki = 226 nM T02551 C1BMD2 44589376 Ki = 0.12 nM T02551 CFB81M 44589377 Ki = 29.2 nM T02551 CS0QD1 44589378 Ki = 658 nM T02551 CP6ZA9 44591012 Ki = 326 nM T02551 C8S1HM 44591042 Ki = 18 nM T02551 CTQ1D6 44591043 Ki = 2874 nM T02551 CZ9I3U 44591044 Ki = 3074 nM T02551 C5C6GE 44591045 Ki = 370 nM T02551 C4YRD3 44591086 Ki = 128 nM T02551 CS5Q7A 44591087 Ki = 335.5 nM T02551 CPA4R6 44591088 Ki = 220 nM T02551 CU37BO 44591098 Ki = 243 nM T02551 CU48CL 44591099 Ki = 67 nM T02551 C7H9SE 44591134 Ki = 50 nM T02551 C6RLW0 44591135 Ki = 50 nM T02551 CBXW20 44591540 Ki = 2454.71 nM T02551 CSO48Z 44591564 Ki > 10000 nM T02551 CYV0C8 44591565 Ki = 3311.31 nM T02551 CH42OK 44591566 Ki > 10000 nM T02551 CT4LV3 44591587 Ki > 10000 nM T02551 C8AY3N 44591605 Ki = 2187.76 nM T02551 CDLR58 44622882 Ki = 0.51 nM T02551 C9N4MQ 44626527 Ki = 3.162 nM T02551 CSJ9F1 44626530 Ki = 1 nM T02551 CCLQ67 44626632 Ki = 5.012 nM T02551 CA93OY 44626637 Ki = 1.585 nM T02551 CPML65 44626639 Ki = 3.981 nM T02551 CDA90T 44626641 Ki = 31.62 nM T02551 C2TBL0 44626734 Ki = 12.59 nM T02551 C7LUV5 44626738 Ki = 1.259 nM T02551 CRCL97 44626740 Ki = 1 nM T02551 CZ25SY 44626744 Ki = 0.631 nM T02551 C5DM7T 44626835 Ki = 1.259 nM T02551 C85ZIF 44626928 Ki = 0.7943 nM T02551 C4BYG5 44626929 Ki = 0.5012 nM T02551 CK5BG2 44626935 Ki = 50.12 nM T02551 CWL84Q 44627022 Ki = 12.59 nM T02551 CGXJ71 44627023 Ki = 0.7943 nM T02551 CBP18J 44627024 Ki = 3.162 nM T02551 C30KEM 44627025 Ki = 0.3981 nM T02551 CV1DO3 44627033 Ki = 1.995 nM T02551 CAH6O1 44627120 Ki = 1 nM T02551 CUE56O 44627123 Ki = 0.3981 nM T02551 CDY32E 44627127 Ki = 0.7943 nM T02551 CJ4ZQ0 44627129 Ki = 6.31 nM T02551 CN1O6P 44627131 Ki = 5.012 nM T02551 CQE59L 44627133 Ki = 0.5012 nM T02551 C4QV9Y 44627238 Ki = 31.62 nM T02551 C1D5FJ 44627240 Ki = 1 nM T02551 CNK4P0 44627242 Ki = 1 nM T02551 CY3LE2 44627245 Ki = 100 nM T02551 C5LN9E 44627351 Ki = 0.2512 nM T02551 CLUN07 44627353 Ki = 1.585 nM T02551 CZ1FY5 44627355 Ki = 0.7943 nM T02551 C3ZWA4 44627357 Ki = 0.5012 nM T02551 CY1TE0 44627358 Ki = 25.12 nM T02551 CG97OK 44627359 Ki = 0.631 nM T02551 C65RAG 44627466 Ki = 10 nM T02551 C06TJC 44627468 Ki = 2.512 nM T02551 CBV8I6 44627470 Ki = 1.259 nM T02551 CR3PL6 44665680 Ki < 1000 nM T02551 CQI0D4 45102707 Ki = 199.53 nM T02551 CSEP-69 45102708 Ki = 630.96 nM T02551 C0DLU3 45109862 IC50 = 334 nM T02551 CQ7D5U 45140376 EC50 = 0.74 nM T02551 CSV08Y 45140377 Ki = 1.28 nM T02551 C98UOH 45260312 Ki = 10 nM T02551 C6Y0LZ 45260341 Ki = 3.162 nM T02551 CHLR80 45260355 Ki = 12.59 nM T02551 C8F1MO 45260357 Ki = 15.85 nM T02551 C31CPA 45260363 Ki = 3.162 nM T02551 CNQ7G1 45260372 Ki = 1.259 nM T02551 C2YL4K 45260377 Ki = 3.981 nM T02551 CXMW87 45260407 Ki = 7.943 nM T02551 C7LRZ1 45260417 Ki = 5.012 nM T02551 CW0X2M 45262323 Ki = 3.162 nM T02551 CQ58RZ 45262339 Ki = 1.259 nM T02551 CE6I0O 45262343 Ki = 1.995 nM T02551 CY87WP 45262345 Ki = 1.259 nM T02551 C6Y4HQ 45262347 Ki = 1.995 nM T02551 C24FEH 45262348 Ki = 3.981 nM T02551 CU03YK 45262349 Ki = 2.512 nM T02551 C3QCD6 45262363 Ki = 1.995 nM T02551 CAT04I 45262369 Ki = 1.585 nM T02551 CY3FD0 45262381 Ki = 1.259 nM T02551 C6PGT0 45262384 Ki = 1.585 nM T02551 C08TZA 45262385 Ki = 6.31 nM T02551 CNE0B7 45262402 Ki = 1.995 nM T02551 CQ29HI 45262403 Ki = 1 nM T02551 C4U7YW 45262404 Ki = 1.259 nM T02551 CF15EW 45262410 Ki = 3.162 nM T02551 CO0HX8 45262412 Ki = 1.259 nM T02551 C08KWJ 45262415 Ki = 1.995 nM T02551 C9FD2N 45262416 Ki = 7.943 nM T02551 CB6KO5 45262417 Ki = 19.95 nM T02551 C1Q9WD 45264008 Ki = 1 nM T02551 C4L3JP 45265219 Ki = 3.162 nM T02551 CR0N7U 45265240 Ki = 2.512 nM T02551 C2A3HT 45265244 Ki = 3.162 nM T02551 CR7UF5 45265257 Ki = 3.981 nM T02551 C5RW2P 45265266 Ki = 3.981 nM T02551 C7N2DT 45265305 Ki = 6.31 nM T02551 C4B6JW 45265589 Ki = 0.7943 nM T02551 C52ALF 45265590 Ki = 2.512 nM T02551 CE2YT8 45265597 Ki = 1.995 nM T02551 CLVE65 45265605 Ki = 1.995 nM T02551 CEUN59 45265612 Ki = 1.259 nM T02551 C4QY5J 45265633 Ki = 3.162 nM T02551 CAHW68 45267251 Ki = 19.95 nM T02551 CW1S6B 45267254 Ki = 2.512 nM T02551 CD47IO 45267261 Ki = 79.43 nM T02551 CJPS81 45267262 Ki = 158.49 nM T02551 C4HOR6 45267270 Ki = 7.943 nM T02551 CM2YT9 45267409 Ki = 67000 nM T02551 CCLR12 45267435 Ki = 6100 nM T02551 CPD18Y 45267471 Ki = 2.512 nM T02551 CL0WP4 45267480 Ki = 2.512 nM T02551 C2H4ZX 45267491 Ki = 0.631 nM T02551 C0KTX2 45267492 Ki = 25.12 nM T02551 C2R9HN 45267503 Ki = 25.12 nM T02551 CEY87M 45267504 Ki = 19.95 nM T02551 CF2R3T 45268112 Ki = 1.259 nM T02551 C3S5ZP 45268113 Ki = 1.585 nM T02551 C0UG9Z 45268119 Ki = 6.31 nM T02551 C37TAV 45268120 Ki = 100 nM T02551 CP1TV2 45268127 Ki = 63.1 nM T02551 C79VFY 45268141 Ki = 5.012 nM T02551 C64NZQ 45268142 Ki = 10 nM T02551 CENZ75 45268148 Ki = 7.943 nM T02551 C71SGH 45268292 Ki = 480 nM T02551 CL0CW7 45268293 Ki = 2700 nM T02551 CM1SA7 45268333 Ki = 158.49 nM T02551 CH53XO 45268345 Ki = 50.12 nM T02551 CHB5U0 45268346 Ki = 158.49 nM T02551 COCN89 45268373 Ki = 50.12 nM T02551 C4MU3C 45268438 Ki = 2.512 nM T02551 CEK21M 45268987 Ki = 15.85 nM T02551 CHB76Z 45268990 Ki = 39.81 nM T02551 CR3YU9 45268999 Ki = 251.19 nM T02551 CW57CP 45269000 Ki = 125.89 nM T02551 CYQ1I7 45269020 Ki = 1 nM T02551 C0F9UT 45269161 Ki = 640 nM T02551 CQP0N3 45269168 Ki = 630 nM T02551 CVH8S4 45269235 Ki = 39.81 nM T02551 CU02ZQ 45269860 Ki = 501.19 nM T02551 CJ18ZC 45270021 Ki = 4200 nM T02551 CF43XE 45270678 Ki = 199.53 nM T02551 CK01NU 45270702 Ki = 39.81 nM T02551 CL42RS 45270813 Ki = 8.5 nM T02551 C5RX4W 45270861 Ki = 22000 nM T02551 CO0P8H 45270903 Ki = 3.162 nM T02551 C7OM4D 45270916 Ki = 125.89 nM T02551 CMQ25P 45271491 Ki = 12.59 nM T02551 CEQ19M 45271499 Ki = 125.89 nM T02551 CESN63 45271510 Ki = 2.512 nM T02551 CMDC23 45271511 Ki = 1.259 nM T02551 C8TXI5 45271516 Ki = 7.943 nM T02551 C5P3FX 45271520 Ki = 3.162 nM T02551 CF9I3G 45271548 Ki = 2.512 nM T02551 C4AJP5 45271653 Ki = 13000 nM T02551 C13RSZ 45271691 Ki = 3100 nM T02551 C6R3LQ 45271737 Ki = 12.59 nM T02551 CM5Q8S 45271738 Ki = 19.95 nM T02551 C42EJD 45271753 Ki = 125.89 nM T02551 CT3DP1 45271760 Ki = 31.62 nM T02551 C5U7LD 45272411 Ki = 501.19 nM T02551 CM9W5B 45272412 Ki = 630.96 nM T02551 CG9CO5 45272414 Ki = 12.59 nM T02551 C4W9NG 45272415 Ki = 158.49 nM T02551 C12WFN 45272425 Ki = 501.19 nM T02551 CK67XC 45272426 Ki = 6.31 nM T02551 CQ2ZS6 45272434 Ki = 3.981 nM T02551 CGKZ21 45272435 Ki = 158.49 nM T02551 CH0MA8 45272437 Ki = 158.49 nM T02551 CW2MD0 45272438 Ki = 158.49 nM T02551 CZ8VO5 45272537 Ki = 3400 nM T02551 CGZW61 45272580 Ki = 1500 nM T02551 CE1P8L 45272616 Ki = 15.85 nM T02551 CEO57P 45272634 Ki = 6.31 nM T02551 CI7C1L 45272635 Ki = 1.585 nM T02551 C9M6XP 45273045 Ki = 44 nM T02551 CIX32S 45273211 EC50 = 1.23 nM T02551 CX1QY9 45273266 Ki = 1.585 nM T02551 C62LGY 45273272 Ki = 63.1 nM T02551 CZ2OL1 45273273 Ki = 125.89 nM T02551 C1YTJ8 45273278 Ki = 199.53 nM T02551 CBM9R2 45273292 Ki = 1.585 nM T02551 CS04AC 45273293 Ki = 125.89 nM T02551 CS95IU 45273334 Ki = 6.31 nM T02551 C19BMF 45273442 Ki = 1300 nM T02551 C7VR4A 45273443 Ki = 330 nM T02551 CFY94G 45273510 Ki = 79.43 nM T02551 CRSF80 45273522 Ki = 1.259 nM T02551 C3DB8P 45273523 Ki = 630.96 nM T02551 CM10UD 45273529 Ki = 100 nM T02551 CRD9C8 45273530 Ki = 125.89 nM T02551 CNQJ09 45273545 Ki = 5.012 nM T02551 C7XC3T 45273551 Ki = 10 nM T02551 CZ71RN 45278805 IC50 = 915 nM T02551 CZN6M7 45278882 IC50 = 1072 nM T02551 CKQG15 45361874 Ki = 1490 nM T02551 CYJ7P8 45379368 Ki > 10000 nM T02551 CU2CA7 45379369 Ki = 42.9 nM T02551 CT3K8Y 45379370 Ki = 513 nM T02551 CT3A1Q 45379373 Ki > 10000 nM T02551 C8TRE1 45379377 Ki > 10000 nM T02551 CML67J 45379515 Ki > 10000 nM T02551 C0SF6L 45482151 Ki = 4.9 nM T02551 CXC65S 45482152 Ki = 320 nM T02551 C8TE2Y 45482153 Ki = 46 nM T02551 C9LX5P 45482169 Ki = 2200 nM T02551 CJD2A3 45482180 Ki = 83 nM T02551 C0CHF4 45482789 IC50 = 660 nM T02551 CLO70J 45483261 Ki = 281.84 nM T02551 C7LD5K 45483269 Ki = 44.67 nM T02551 CO1M6P 45483654 Ki = 230 nM T02551 CIV3Q4 45483655 Ki = 70 nM T02551 C9D0RB 45486325 EC50 = 0.493 nM T02551 CD2OP0 45486328 EC50 = 0.528 nM T02551 C75KWB 45486329 Ki = 0.685 nM T02551 C41IVO 45486330 EC50 = 0.52 nM T02551 CPSV53 45486332 Ki = 2.65 nM T02551 C8NS2H 45486333 Ki = 4.78 nM T02551 C5BR3T 45486336 Ki = 1.27 nM T02551 CCVJ58 45486341 Ki = 0.441 nM T02551 CLK12R 45486360 Ki = 0.4 nM T02551 CU5LO4 45486363 Ki = 0.435 nM T02551 C9G1TW 45486364 Ki = 0.19 nM T02551 CSQ1J5 45487336 Ki = 63.1 nM T02551 C24WVU 45487513 Ki = 50.12 nM T02551 CK9EC3 46180160 Ki = 0.186 nM T02551 CLBT94 46190877 Ki = 5011.87 nM T02551 COFU37 46225335 Ki > 10000 nM T02551 C9XTG3 46225336 Ki > 10000 nM T02551 C96LBQ 46225337 Ki > 10000 nM T02551 C6MC8Z 46225569 Ki = 501.19 nM T02551 CS6Y9W 46225581 Ki = 1584.89 nM T02551 C78DON 46225582 Ki > 10000 nM T02551 CC8E3T 46225583 Ki = 3981.07 nM T02551 CML42B 46225584 Ki = 1584.89 nM T02551 CY7NM6 46227242 Ki > 10000 nM T02551 CR9S7B 46227243 Ki > 10000 nM T02551 C9A8FV 46227273 Ki > 10000 nM T02551 CL3KU2 46227284 Ki > 10000 nM T02551 CS4O6A 46227317 Ki = 251 nM T02551 CE1L6H 46227320 Ki > 10000 nM T02551 CSQ9D5 46227325 Ki > 10000 nM T02551 C9FV8B 46233097 Ki = 5.57 nM T02551 C24GSH 46233135 Ki = 3.71 nM T02551 C5TC2S 46830335 IC50 > 10000 nM T02551 C1K7FL 46830336 IC50 > 10000 nM T02551 C1N4KX 46842383 IC50 > 10000 nM T02551 C0WJ5L 46850462 Ki = 1300 nM T02551 CN3RH6 46850464 Ki = 280 nM T02551 CC62SX 46866711 IC50 = 1195 nM T02551 C03LTM 46869265 Ki = 210 nM T02551 CK8A1O 46880462 Ki > 10000 nM T02551 C9KDP4 46880463 Ki > 10000 nM T02551 CODR73 46880498 Ki > 10000 nM T02551 CHJ5Y6 46880566 Ki > 10000 nM T02551 CE9PG2 46880567 Ki > 10000 nM T02551 C01PGO 46880568 Ki > 10000 nM T02551 CS7L4X 46880569 Ki > 10000 nM T02551 C0PXY7 46880628 Ki > 10000 nM T02551 CD37LU 46880629 Ki > 10000 nM T02551 CUY89F 46880630 Ki > 10000 nM T02551 C4P6XS 46880631 Ki > 10000 nM T02551 CJ53KF 46880672 Ki > 10000 nM T02551 CYJC08 46880673 Ki > 10000 nM T02551 C1RI9O 46880674 Ki > 10000 nM T02551 CM2ZY5 46881408 Ki = 25.12 nM T02551 C1R8WT 46881409 Ki = 79.43 nM T02551 CT2VZ3 46881410 Ki > 630.96 nM T02551 CW62EC 46881411 Ki > 630.96 nM T02551 CAHF16 46881412 Ki = 316.23 nM T02551 CT9IF0 46881413 Ki = 125.89 nM T02551 C2MC4K 46881463 Ki = 3.981 nM T02551 C27IES 46881464 Ki > 630.96 nM T02551 CP24SO 46881465 Ki > 630.96 nM T02551 C4Y9UE 46881466 Ki = 0.2512 nM T02551 C9AJI3 46881467 Ki > 630.96 nM T02551 C0EF4O 46882004 Ki = 5.012 nM T02551 CR4CN8 46882005 Ki = 3.981 nM T02551 CR9SO6 46882006 Ki = 79.43 nM T02551 CJMC05 46882007 Ki = 1.585 nM T02551 CJYU26 46882008 Ki > 630.96 nM T02551 CAU9M8 46882009 Ki = 79.43 nM T02551 CB34TO 46882049 Ki = 125.89 nM T02551 CDTA05 46882050 Ki = 50.12 nM T02551 CB13IH 46882051 Ki = 1 nM T02551 C0HM3E 46882052 Ki = 63.1 nM T02551 CM93UE 46882053 Ki = 15.85 nM T02551 CDXI13 46882054 Ki = 251.19 nM T02551 C4BH9E 46882458 Ki = 3.981 nM T02551 CF8IJ2 46882520 Ki = 100 nM T02551 CQN87I 46882521 Ki = 31.62 nM T02551 C56ULO 46882522 Ki = 19.95 nM T02551 CX72IN 46882583 Ki = 630.96 nM T02551 CB8GE1 46884818 IC50 > 10000 nM T02551 C4MQ0A 46884856 IC50 > 10000 nM T02551 CCNT25 46884898 IC50 > 10000 nM T02551 C3MSG2 46885027 IC50 > 10000 nM T02551 CB7XI0 46885213 IC50 > 10000 nM T02551 CRW2I9 46893146 Ki = 0.12 nM T02551 CV9E5Y 46912547 Ki = 87.6 nM T02551 C34ILU 46912548 Ki = 100 nM T02551 CGSN70 46917563 Ki = 0.71 nM T02551 CEH10Y 46917637 Ki = 1.2 nM T02551 C7FX8L 46931072 Ki = 95 nM T02551 CKO76R 46931815 Ki = 0.631 nM T02551 CUTX67 46934428 IC50 = 248 nM T02551 CYWX19 49780808 Ki = 50.12 nM T02551 C9RI3L 49780809 Ki = 3.981 nM T02551 C39KWP 49781039 Ki = 251.19 nM T02551 C9O2RB 49781040 Ki = 3.162 nM T02551 C7T3KS 49781255 Ki = 5.012 nM T02551 CYL65E 49781476 Ki = 10 nM T02551 CFQN89 49781477 Ki = 50.12 nM T02551 CL82ES 49781478 Ki = 6.31 nM T02551 CESC01 49782398 Ki = 53 nM T02551 C8BWU1 49782600 Ki = 27 nM T02551 C6I0NJ 49782601 Ki = 17 nM T02551 C20CVH 49782602 Ki = 38 nM T02551 CY4FW1 49782603 Ki = 73 nM T02551 CXJ59F 49782604 Ki = 280 nM T02551 CD9ZH7 49782836 Ki = 9.9 nM T02551 CL1J4C 49782837 Ki = 410 nM T02551 CB53QP 49782841 Ki = 1.6 nM T02551 CENR09 49783039 Ki = 2.5 nM T02551 CZ5G9J 49783040 Ki = 4.7 nM T02551 C98JVY 49783041 Ki = 4 nM T02551 CRML65 49783042 Ki = 28 nM T02551 COM8D5 49798797 Ki = 1585 nM T02551 C9ZYH8 49798799 Ki = 4938 nM T02551 C4TXW8 49798812 Ki = 49 nM T02551 C9KOV8 49798833 Ki = 142 nM T02551 C6LP9T 49798835 Ki = 10.9 nM T02551 C6RE1F 49798837 Ki = 11.2 nM T02551 CMQ23B 49798839 Ki = 3 nM T02551 C2WZ9Y 49798853 Ki = 46.7 nM T02551 CU34RI 49798855 Ki = 2.1 nM T02551 CM86YK 49798857 Ki = 9.3 nM T02551 CTDN46 49798874 Ki = 0.9 nM T02551 CO4K6F 49798877 Ki = 250 nM T02551 C69EKV 49798878 Ki = 204 nM T02551 CWQ9Y1 49798879 Ki = 96.9 nM T02551 CV1S3H 49799687 Ki = 94.4 nM T02551 CBR67S 49799691 Ki = 2927 nM T02551 C5A6TG 49799693 Ki = 188 nM T02551 CZ8A2G 49799695 Ki = 132 nM T02551 CCV35T 49799709 Ki = 849 nM T02551 CLY02B 49799713 Ki = 68.2 nM T02551 CDTS15 49799715 Ki = 2983 nM T02551 CDAB96 49836026 Ki = 7.943 nM T02551 C4R2YS 49850567 Ki = 79.43 nM T02551 C07JTU 49850570 Ki = 125.89 nM T02551 CK68QR 49850672 Ki = 100 nM T02551 CN5XR1 49850772 Ki = 50.12 nM T02551 CR4EZ0 49850870 Ki = 199.53 nM T02551 C5K4EC 49850872 Ki = 158.49 nM T02551 C8AW0R 49850874 Ki = 100 nM T02551 C9KIU1 49864289 IC50 = 1426 nM T02551 CHO9C0 49864292 IC50 = 943 nM T02551 C5O7HP 49864396 Ki = 842 nM T02551 C90MTG 49864602 IC50 = 2893 nM T02551 C5BCS4 49864722 IC50 = 2416 nM T02551 CKZO79 49864723 IC50 = 2508 nM T02551 C74LZS 49864724 IC50 = 1171 nM T02551 CKWA93 49865589 Ki = 79.43 nM T02551 C8J5PI 49865599 Ki = 198 nM T02551 CP63AX 49865600 Ki = 25 nM T02551 CA1IY0 49865601 Ki = 198 nM T02551 CXWL20 49865623 Ki = 3.981 nM T02551 CC5KD7 49865639 Ki = 133 nM T02551 C1B5RD 49865640 Ki = 383 nM T02551 C51PJT 49865641 Ki = 207 nM T02551 C3KF6B 49865668 Ki = 1 nM T02551 C2RY0J 50878551 Ki = 489.78 nM T02551 C1W6TV 50898777 Ki > 10000 nM T02551 CXMZ73 50898778 Ki > 10000 nM T02551 C8TA1J 51003550 IC50 = 1520 nM T02551 CQ1UJ7 51003551 IC50 = 482 nM T02551 CGMI37 51003586 IC50 = 623 nM T02551 CE4KP1 51050257 Ki > 10000 nM T02551 C2HGK8 51122451 Ki = 4 nM T02551 CMYT24 51353673 Ki = 6.2 nM T02551 C5W4PN 51353674 Ki = 10.9 nM T02551 C0UBA8 51353675 Ki = 13.8 nM T02551 CU3C4O 51353676 Ki = 0.65 nM T02551 CB3A9S 51353677 Ki = 6.9 nM T02551 C1LHZ4 51353678 Ki = 0.52 nM T02551 CIO10J 51353988 Ki = 2.5 nM T02551 CWFU41 51353989 Ki = 0.17 nM T02551 CA01KY 51353990 Ki = 5.2 nM T02551 CA8E9Q 51353991 Ki = 3.6 nM T02551 CW8LE6 51353992 Ki = 1.1 nM T02551 CL8WR0 51354273 Ki = 8.4 nM T02551 CW03GI 51354274 Ki = 19.6 nM T02551 C2DG1Z 51354275 Ki = 1.1 nM T02551 CT8MC6 51354277 Ki = 1.1 nM T02551 CEL30Q 51354279 Ki = 24.9 nM T02551 CU9B6W 51354566 Ki = 6.2 nM T02551 COD5H3 51354851 Ki = 4.2 nM T02551 CPN8T3 51354853 Ki = 18.2 nM T02551 C7Q2MW 51355139 Ki = 18.5 nM T02551 CMYZ04 51355143 Ki = 13.6 nM T02551 C42GMN 52937680 Ki = 0.55 nM T02551 CZ06OU 52937773 Ki = 330 nM T02551 CYC05D 52937774 Ki = 44 nM T02551 C96LHK 52937776 Ki = 0.71 nM T02551 C30RKG 52937777 Ki = 0.59 nM T02551 C78FZD 52937871 Ki = 39 nM T02551 C1S9VT 52937875 Ki = 6.3 nM T02551 CFK1D4 52937876 EC50 = 0.0028 nM T02551 CIWA18 52938727 Ki = 1.14 nM T02551 C6XY8V 52938728 Ki = 2.67 nM T02551 CY2SH8 52939845 Ki = 1.9 nM T02551 C7U0IC 52939846 Ki = 250 nM T02551 CJ19FP 52940753 Ki = 6.31 nM T02551 CCDZ51 52940788 Ki = 10 nM T02551 C2RW5A 52940961 Ki = 3.981 nM T02551 CS5I2W 52940985 Ki = 290 nM T02551 CCK37R 52941006 EC50 = 0.25 nM T02551 C8FZL4 52941427 Ki = 39.81 nM T02551 C09RJS 52943802 Ki = 420 nM T02551 CQJ7C0 52945023 Ki = 31.62 nM T02551 CT51OC 52945819 Ki = 76 nM T02551 COZ9J3 52946432 Ki = 158.49 nM T02551 C19ZKQ 52946556 Ki = 52.5 nM T02551 CI5V3X 52947507 Ki = 158.49 nM T02551 C6ZSQ8 52947516 Ki = 12.59 nM T02551 CN32PV 52947694 Ki = 3.981 nM T02551 CUV0G4 52947756 Ki = 4.2 nM T02551 CZ01DH 52948653 Ki = 125.89 nM T02551 C9OSI0 52949300 Ki = 3.981 nM T02551 C4IV2J 53248158 Ki = 20.5 nM T02551 C03JEZ 53248159 Ki = 6.2 nM T02551 C2G0ZY 53248208 Ki = 28.6 nM T02551 C2UKM3 53248209 Ki = 5.4 nM T02551 C8KW9J 53248210 Ki = 13.9 nM T02551 C87SLP 53248211 Ki = 8 nM T02551 CVD7E5 53248212 Ki = 9.5 nM T02551 CX6KG9 53248213 Ki = 4 nM T02551 C63MQD 53248256 Ki = 10.1 nM T02551 CG2O7F 53248257 Ki = 2.6 nM T02551 CRK87G 53248258 Ki = 3.8 nM T02551 C73WQX 53248259 Ki = 2.9 nM T02551 CKOV84 53248260 Ki = 4.6 nM T02551 C09IXA 53248261 Ki = 1.5 nM T02551 C5K7NT 53248298 Ki = 6.1 nM T02551 C28DOY 53248299 Ki = 38.6 nM T02551 CIM15A 53248300 Ki = 4.8 nM T02551 C0LS5Y 53248345 Ki = 71.5 nM T02551 CSU1D5 53248346 Ki = 129 nM T02551 CBS3U2 53248347 Ki = 80.8 nM T02551 C85RJF 53248348 Ki = 104 nM T02551 CF3AO9 53248349 Ki = 134 nM T02551 CSF8M1 53248393 Ki = 467 nM T02551 C6P5WJ 53248394 Ki = 162 nM T02551 CN4SY6 53248395 Ki = 393 nM T02551 CC78FG 53248673 Ki = 13.5 nM T02551 CL3WJ1 53248675 Ki = 5.4 nM T02551 CG6T2N 53248677 Ki = 2.7 nM T02551 C5C8ZN 53317208 Ki = 8.14 nM T02551 CSM53O 53317282 Ki = 9.18 nM T02551 C8JO1K 53317511 Ki > 10000 nM T02551 C68UVE 53317620 Ki = 8.16 nM T02551 CKXS49 53317727 Ki = 890 nM T02551 C36MWP 53318500 Ki = 35 nM T02551 CA31DT 53318564 Ki = 102 nM T02551 CU4CR9 53318565 Ki = 189 nM T02551 C61DNP 53320009 IC50 = 1300 nM T02551 C9ZDR5 53320010 IC50 = 2922 nM T02551 CM5N9H 53320353 Ki > 10000 nM T02551 CODA90 53320569 Ki = 7155 nM T02551 CI1G0L 53321123 Ki = 2400 nM T02551 C5DL8F 53321194 Ki = 23.4 nM T02551 C3M6UO 53322449 Ki = 21 nM T02551 CHU18S 53322522 Ki = 8 nM T02551 CQLK01 53322638 IC50 = 180 nM T02551 CZ5AN7 53322729 Ki > 10000 nM T02551 C0WT8G 53322769 Ki = 1.1 nM T02551 C2V5SI 53323810 Ki = 191 nM T02551 CD78CH 53323858 Ki = 4514 nM T02551 C3B4SQ 53323859 Ki = 1.82 nM T02551 C32YWL 53324045 Ki = 62 nM T02551 CR4W9L 53324553 Ki = 5215 nM T02551 CP7MR3 53325130 Ki = 281 nM T02551 C35GJZ 53325137 Ki = 19.9 nM T02551 CB6RV7 53325138 Ki = 7.7 nM T02551 CRQF15 53325242 Ki = 209 nM T02551 CB37XF 53325861 Ki > 10000 nM T02551 CLPK26 53326377 Ki = 539 nM T02551 CIR65P 53326378 Ki = 44 nM T02551 C0UC1W 53326601 Ki = 0.8 nM T02551 CQ8I3D 53326670 Ki = 230 nM T02551 CS5Z7X 53327908 Ki = 0.12 nM T02551 C5TVA7 53359024 Ki > 10000 nM T02551 CLZ09P 53359025 Ki = 1958 nM T02551 CPQ1E2 53361301 Ki = 84 nM T02551 CABK98 53361302 Ki = 610 nM T02551 CK0M7F 53363109 Ki = 320 nM T02551 CG24FV 53363110 Ki = 590 nM T02551 C28MPE 53363199 Ki = 440 nM T02551 CN3C4E 53363200 Ki = 250 nM T02551 CYW7M4 53363201 Ki = 220 nM T02551 C6EU7I 53363202 Ki = 100 nM T02551 CMI25H 53364083 Ki = 230 nM T02551 C1UWI5 53364153 Ki = 31 nM T02551 C78PUJ 53364154 Ki = 96 nM T02551 CRB76A 53364155 Ki = 74 nM T02551 CZV06L 53364225 Ki = 36 nM T02551 CQ7PX0 53364226 Ki = 61 nM T02551 CCA02T 53364227 Ki = 72 nM T02551 CEIG81 53391632 Ki > 20000 nM T02551 CQ3M2A 53391731 Ki > 15000 nM T02551 CMOZ61 53475319 EC50 = 1.7 nM T02551 C0JC2O 54325398 Ki = 0.7943 nM T02551 CX7H3P 54325399 Ki = 3.981 nM T02551 CV2G4S 54437013 Ki = 15.85 nM T02551 C5JL8O 54437014 Ki = 3.981 nM T02551 CL5QO2 54493650 Ki = 7.943 nM T02551 CCM43W 54580387 Ki = 101 nM T02551 CKND43 54580905 Ki = 0.25 nM T02551 CF6G4L 54580906 Ki = 0.21 nM T02551 CHNI24 54581963 Ki = 0.27 nM T02551 CM5TK0 54581964 Ki = 0.29 nM T02551 CX6EI5 54582316 Ki = 2.7 nM T02551 C8AT1S 54583897 Ki = 1.6 nM T02551 CW9Z2J 54583898 Ki = 0.5 nM T02551 CN6O2E 54584336 Ki = 67.9 nM T02551 CFPM39 54585226 Ki = 1 nM T02551 CIMS79 54585306 Ki = 0.8 nM T02551 CCO81W 54585447 Ki = 0.25 nM T02551 CL23NI 54585810 Ki = 12 nM T02551 CW1I5B 54585811 Ki = 1.3 nM T02551 C3QJP1 54735210 Ki = 1.1 nM T02551 CL5I1R 54753271 Ki = 544 nM T02551 CY27RS 56360144 EC50 = 105 nM T02551 CF59RX 56361674 EC50 = 151 nM T02551 CQ3AR0 56589560 Ki = 304 nM T02551 C4XGR3 56589561 Ki = 4676 nM T02551 C9PHZ3 56594402 Ki > 10000 nM T02551 C82IVX 56594533 Ki > 10000 nM T02551 CT4J5C 56594534 Ki = 681 nM T02551 CG0K6E 56597637 Ki = 8.511 nM T02551 CJ57IF 56658006 Ki = 574 nM T02551 CTWV58 56658008 Ki = 3.8 nM T02551 C1CJ8P 56664948 Ki = 879 nM T02551 C26RNX 56664950 Ki = 785 nM T02551 CRPA72 56664952 Ki = 7 nM T02551 CW7F5G 56675269 Ki = 930 nM T02551 CC2B8F 56678599 Ki = 1536 nM T02551 C28ECA 56681925 Ki = 427 nM T02551 CLX25U 56681927 Ki = 251 nM T02551 CFE60O 56833378 Ki = 1.8 nM T02551 C04VKH 56833379 Ki = 12 nM T02551 CAS80D 56833463 Ki = 2 nM T02551 CUXP15 56833464 Ki = 2 nM T02551 C6DEW7 56837419 Ki = 0.23 nM T02551 CZ1WY0 56837634 Ki = 0.44 nM T02551 CKJ2U0 56837635 Ki = 0.3 nM T02551 CZP6E4 56837636 Ki = 11 nM T02551 CXJ7R9 56926585 Ki = 5900 nM T02551 CH1S9B 56926586 Ki = 4200 nM T02551 CJ42HS 56926587 Ki = 17000 nM T02551 C7G5PJ 56941366 EC50 = 0.1 nM T02551 CB0P9N 56944383 Ki = 1.1 nM T02551 C1TC7Q 56963799 Ki > 10000 nM T02551 CD9I4N 57334553 IC50 = 24.8 nM T02551 C6H9UV 57345617 Ki = 9.7 nM T02551 CZU6L2 57345618 Ki = 208.8 nM T02551 CK9G8H 57345619 Ki = 3043 nM T02551 CU2M7Q 57345620 Ki = 16 nM T02551 C6QAE5 57383397 Ki = 880 nM T02551 C0KR7X 57383401 Ki = 350 nM T02551 C6NCE0 57383405 Ki = 370 nM T02551 CQO45V 57383408 Ki > 50000 nM T02551 C7XJ1A 57383414 Ki = 130 nM T02551 CMW19O 57383430 Ki = 230 nM T02551 CL8N9J 57383431 Ki = 9200 nM T02551 CT5O6F 57383434 Ki = 3400 nM T02551 C7LQV0 57383436 Ki = 21000 nM T02551 C0QM2U 57390115 Ki = 4.9 nM T02551 CZ12PI 57390116 Ki = 0.61 nM T02551 CRG2X7 57390117 Ki = 330 nM T02551 CR9L2W 57390118 Ki = 0.88 nM T02551 C26DAH 57390119 Ki = 100 nM T02551 CATM39 57390694 Ki = 863 nM T02551 C6S0IE 57390695 Ki = 1051 nM T02551 CV08WY 57391216 Ki = 68 nM T02551 CD75YK 57391306 Ki = 243 nM T02551 C07PMA 57391307 Ki = 885 nM T02551 C0T9UH 57391895 Ki = 83 nM T02551 CPN87T 57391896 Ki = 11 nM T02551 C64AWK 57391897 Ki = 78 nM T02551 CWT20M 57393083 Ki = 262 nM T02551 C1M4PZ 57393627 Ki = 350 nM T02551 C7E4BW 57393628 Ki = 0.34 nM T02551 CGWK23 57393634 Ki = 110 nM T02551 CADH19 57394285 Ki = 1020 nM T02551 C0WA3H 57394810 Ki = 130 nM T02551 C39YHG 57395340 Ki = 16 nM T02551 C35RST 57395341 Ki = 160 nM T02551 CD4A3P 57396484 Ki = 778 nM T02551 C4EXS6 57396571 Ki = 726 nM T02551 C3GW6L 57398351 Ki = 696 nM T02551 CO50ZB 57398352 Ki = 544 nM T02551 C5YZM2 57398875 Ki = 10 nM T02551 CJ41PW 57399432 Ki = 152 nM T02551 CO3B4P 57399494 Ki = 590 nM T02551 CI9XS8 57400556 Ki = 0.66 nM T02551 C20IPH 57400557 Ki = 1.2 nM T02551 CU0C3D 57400562 Ki = 930 nM T02551 CZX05B 57401706 Ki = 160 nM T02551 CYN38R 57401819 Ki = 261 nM T02551 CO0XD2 57401820 Ki = 422 nM T02551 CO04CI 57402365 Ki = 170 nM T02551 C27OEI 57402366 Ki = 0.5 nM T02551 CFJ27E 57402787 Ki = 3.5 nM T02551 C92HON 57402951 Ki = 777 nM T02551 CX0B5M 57403525 Ki = 666 nM T02551 CWBG94 57403981 Ki = 13 nM T02551 CQB6F9 57456630 Ki = 45 nM T02551 C9PLU4 57527911 Ki > 100000 nM T02551 CH3T2M 57587922 Ki = 185 nM T02551 C0M5PN 57873490 Ki = 560 nM T02551 CH1BN8 57873491 Ki = 159 nM T02551 CI5UO1 57873492 Ki = 40 nM T02551 C2D9HA 57873499 Ki = 40 nM T02551 C81MLX 57873504 Ki = 186 nM T02551 C7L9IE 57873508 Ki = 46 nM T02551 CZRL39 57873513 Ki = 14 nM T02551 C98WTS 57873515 Ki = 24 nM T02551 C6BHT3 57873518 Ki = 61 nM T02551 CPX17D 57873520 Ki = 0.9 nM T02551 C54ROE 57873522 Ki = 12 nM T02551 CM7PI1 57873525 Ki = 73 nM T02551 CMUR21 57873527 Ki = 122 nM T02551 CO5Y9Q 57873531 Ki = 0.4 nM T02551 CCX12B 58358826 Ki = 1.9 nM T02551 C2AY1P 60148494 EC50 = 0.26 nM T02551 CIFJ86 60148495 EC50 = 0.56 nM T02551 CHJL24 60148496 EC50 = 0.87 nM T02551 CEY2I7 60148497 EC50 = 1.26 nM T02551 C4MV2N 60149678 Ki = 15700 nM T02551 C2Q5VD 60165416 Ki = 31 nM T02551 C9JL3F 60165418 Ki = 100 nM T02551 C9Q7MR 60165801 EC50 = 0.26 nM T02551 C5RUP6 60167166 Ki = 214 nM T02551 CRH49P 60167309 Ki = 288.4 nM T02551 COHK72 60167451 Ki = 63.1 nM T02551 C30SVG 60167452 Ki = 17.78 nM T02551 C6EU1T 60194424 EC50 = 1.5 nM T02551 CI30FT 60204111 Ki = 1.7 nM T02551 CWSA08 60204112 Ki = 27 nM T02551 CXI15A 60481587 EC50 > 50000 nM T02551 C3XL7O 66561967 Ki > 10000 nM T02551 CG5BP2 66574145 IC50 = 0.6 nM T02551 CMG51Y 68807656 Ki = 152 nM T02551 C34GMW 69599704 Ki = 2.4 nM T02551 CQH61C 70681318 Ki = 15 nM T02551 CT38JR 70683414 Ki = 1570 nM T02551 C6PD9Q 70684338 Ki = 21000 nM T02551 CTHV58 70684339 Ki = 11000 nM T02551 CB9V3R 70686493 Ki = 1770 nM T02551 C1P3GF 70686494 Ki = 36000 nM T02551 C3V5QJ 70686495 Ki = 7930 nM T02551 C2U6KV 70688594 Ki = 36000 nM T02551 CG80JF 70690651 Ki = 13200 nM T02551 CZH6F9 70690652 Ki = 2140 nM T02551 C6TJA5 70690653 Ki = 1500 nM T02551 CPO08R 70691861 Ki = 120 nM T02551 CD37EI 70691866 Ki = 524 nM T02551 CU82LJ 70692801 Ki = 11000 nM T02551 C18ETD 70692802 Ki = 8800 nM T02551 C98YAU 70696888 Ki = 5300 nM T02551 CC43QK 71151588 Ki = 0.1 nM T02551 C2AQ7H 71195187 Ki > 1000 nM T02551 C0O5KW 71449034 Ki = 1850 nM T02551 CX17SY 71449211 EC50 = 4.3 nM T02551 CSC3R7 71450213 Ki = 1148 nM T02551 CE6YD5 71450707 Ki = 460 nM T02551 CBP03H 71450812 Ki = 83 nM T02551 CDI84E 71450922 IC50 > 10000 nM T02551 C08KHB 71452040 EC50 = 32.2 nM T02551 C0XW8E 71452041 Ki = 282 nM T02551 CTDN12 71452341 Ki = 6739 nM T02551 CE0R9D 71454275 Ki = 2520 nM T02551 C4X9KY 71454294 Ki = 350 nM T02551 CA65OQ 71454295 Ki = 33 nM T02551 C8YKT4 71454405 Ki = 220 nM T02551 CQMK12 71454927 Ki = 50 nM T02551 CD4HQ6 71456045 Ki = 580 nM T02551 CD78KL 71456046 Ki = 390 nM T02551 CDSX56 71457372 Ki = 1147 nM T02551 CSX5J0 71457844 Ki = 160 nM T02551 CNM83V 71457956 Ki = 75 nM T02551 CNQ5B6 71458040 Ki = 180 nM T02551 C84QJC 71458071 Ki = 720 nM T02551 C3X1ZG 71459659 EC50 = 0.53 nM T02551 CH5YG1 71459660 EC50 = 0.94 nM T02551 CI6OW4 71459759 Ki = 210 nM T02551 CSY3U1 71459760 Ki = 370 nM T02551 CD10CQ 71459761 Ki = 85 nM T02551 CYGO39 71459901 Ki = 0.1995 nM T02551 CG0WO9 71459954 Ki > 5000 nM T02551 C9ESJ4 71461481 Ki = 370 nM T02551 C9VE0P 71462090 Ki = 1.1 nM T02551 CKX5O8 71463061 Ki = 5466 nM T02551 C82GIQ 71463207 Ki = 530 nM T02551 CE92DF 71528209 Ki = 1492 nM T02551 C5PHM9 71571370 EC50 = 4400 nM T02551 CS0FY1 71571378 EC50 = 530 nM T02551 CUN24P 71571394 EC50 = 278 nM T02551 CE13MV 71571401 EC50 = 9700 nM T02551 CDU24A 71571402 EC50 = 310 nM T02551 C83LQO 71571413 EC50 = 2600 nM T02551 C0M7QU 71571423 EC50 = 310 nM T02551 C1Z2OC 71571433 EC50 = 98 nM T02551 CRMC90 71571436 EC50 = 548 nM T02551 CNQ2J1 71575525 Ki = 4700 nM T02551 CO3E4N 71583848 Ki = 20 nM T02551 C8N2ML 71583849 Ki = 18 nM T02551 CO4P6L 71604368 EC50 = 17 nM T02551 CWAO49 71604376 EC50 = 115 nM T02551 CJCO20 71604380 EC50 = 9300 nM T02551 C5VH2Z 71657942 Ki = 3.9 nM T02551 CY9ES0 71657943 Ki = 2.9 nM T02551 CU41CZ 71657944 Ki = 5.5 nM T02551 C0S6YV 71657945 Ki = 9 nM T02551 CX52VK 71657946 Ki = 1.8 nM T02551 C6KJW5 71657947 Ki = 3.7 nM T02551 C6AQG0 71658072 Ki = 8.8 nM T02551 CQ3W7X 71658073 Ki = 7.5 nM T02551 CE3V4J 71658074 Ki = 2.5 nM T02551 C40XRK 71658075 Ki = 1.5 nM T02551 CPI8E9 71658076 Ki = 9 nM T02551 CC1U6V 71658077 Ki = 13.2 nM T02551 C8LX4D 71658203 Ki = 11.6 nM T02551 CVX3G1 71658204 Ki = 4.8 nM T02551 C29STX 71658205 Ki = 8 nM T02551 CR0EN8 71658206 Ki = 15 nM T02551 CF41PZ 71658207 Ki = 17.9 nM T02551 C7LMV3 71658208 Ki = 44.2 nM T02551 CIAR53 71658338 Ki = 7.2 nM T02551 CZ65JA 71659909 Ki = 0.7 nM T02551 C8PLQ7 71660285 EC50 = 30.3 nM T02551 CW35XI 71722291 Ki = 130 nM T02551 C4EC8K 71722293 Ki = 23 nM T02551 C4FJV9 71722295 Ki = 55 nM T02551 C8H5OT 71722297 Ki = 17 nM T02551 C3SDV1 71722299 Ki = 28 nM T02551 CY4NH1 71722300 Ki = 53 nM T02551 CTI15V 71724940 EC50 = 80 nM T02551 CGH7I1 71724941 EC50 = 160 nM T02551 C24SVN 71724943 EC50 = 13.3 nM T02551 C64GLV 71724944 EC50 = 3 nM T02551 CB3WQ5 71724946 EC50 = 50 nM T02551 CG34PQ 71724947 EC50 = 37.6 nM T02551 CF0TW3 71724948 EC50 = 520 nM T02551 CV5OH2 71724949 EC50 = 576 nM T02551 CKP3M7 71724951 EC50 = 42 nM T02551 CUB76P 71724952 EC50 = 6.9 nM T02551 CE4A7V 71724954 EC50 = 192 nM T02551 CD53XP 71724955 EC50 = 411 nM T02551 CLTX37 71724956 EC50 = 710 nM T02551 C4YA9Q 71724957 EC50 = 130 nM T02551 C9C2IE 71724959 EC50 = 4.4 nM T02551 CDW76R 71724960 EC50 = 116 nM T02551 C1BYT9 71724961 EC50 = 563 nM T02551 C3TAK6 71724962 EC50 = 980 nM T02551 CI0D9X 71724963 EC50 = 510 nM T02551 C2I1ML 71724964 EC50 = 6.4 nM T02551 C9P2RK 71724965 EC50 = 208 nM T02551 C0X8AZ 71724966 EC50 = 33 nM T02551 CBIF31 71724967 EC50 = 33 nM T02551 C2LI5P 71724968 EC50 = 200 nM T02551 CH6C3U 71724969 EC50 = 2100 nM T02551 CI3V7S 71724970 EC50 = 63 nM T02551 CC08MW 71724971 EC50 = 13.5 nM T02551 CZIH39 71724974 EC50 = 118 nM T02551 CD2U5X 71724975 EC50 = 45 nM T02551 CPIC98 71724976 EC50 = 25.7 nM T02551 CXM9B5 71724977 EC50 = 810 nM T02551 CM63QP 71724978 EC50 = 59 nM T02551 C6C9IT 71724979 EC50 = 2800 nM T02551 CQRY07 71724980 EC50 = 98 nM T02551 CJS8I1 71724983 EC50 = 3800 nM T02551 CC7T2D 71724985 EC50 = 13 nM T02551 CC5FG2 71724986 EC50 = 266 nM T02551 CV09TJ 71724987 EC50 = 7 nM T02551 CIX5F7 71724989 EC50 = 167 nM T02551 C14LXP 71724991 EC50 = 9.5 nM T02551 CUFB92 71724993 EC50 = 473 nM T02551 CFS28E 71724994 EC50 = 33.8 nM T02551 C0F2WP 71724995 EC50 = 4.3 nM T02551 CEJ2L9 71724996 EC50 = 81 nM T02551 CQL6U0 71724997 EC50 = 997 nM T02551 C4NIK3 71725006 EC50 = 1900 nM T02551 CM31ZP 71725009 EC50 = 472 nM T02551 C8HQP2 71725014 EC50 = 630 nM T02551 CR6JF2 71725020 EC50 = 126 nM T02551 C0X4CR 71725021 EC50 > 100000 nM T02551 C6MTL4 71725024 EC50 = 41 nM T02551 C8URA5 71725025 EC50 = 210 nM T02551 CFY64I 71725026 EC50 = 1600 nM T02551 C09ZBK 71725027 EC50 = 610 nM T02551 CEZN65 71725031 EC50 = 284 nM T02551 CXA9N4 71725039 EC50 = 290 nM T02551 CCWP92 71725040 EC50 = 1300 nM T02551 CZ2MG4 71725047 EC50 = 5 nM T02551 C54VLH 71725049 EC50 = 114 nM T02551 C9HWI1 71725050 EC50 = 2900 nM T02551 C3V6XP 71725052 EC50 = 285 nM T02551 CRV8K6 71725061 EC50 = 1900 nM T02551 CEQL80 71725064 EC50 = 280 nM T02551 C7HKL3 71725065 EC50 = 60.9 nM T02551 CQO30I 71733932 Ki = 0.12 nM T02551 C93QMB 71733935 Ki = 0.17 nM T02551 COM72V 71734028 Ki = 3.2 nM T02551 C4S5WD 71734029 Ki = 8.6 nM T02551 C2ZX1W 71734031 Ki = 0.24 nM T02551 C7GDW5 71734126 Ki = 10 nM T02551 CQJ8P4 71734127 Ki = 10 nM T02551 CR53GT 71734129 Ki = 0.43 nM T02551 C31THM 72164180 Ki = 44.5 nM T02551 C56VLM 72164181 Ki > 10000 nM T02551 CD8A9K 72164182 Ki = 62 nM T02551 C4C0BH 72164183 Ki = 221 nM T02551 CQU81Y 72164299 Ki = 41 nM T02551 CF0H7K 72164300 Ki = 92 nM T02551 C7WM5U 72164301 Ki = 41 nM T02551 C4HO2U 72164302 Ki = 123 nM T02551 C08NOR 72187659 EC50 = 32 nM T02551 CQ70NJ 72187662 EC50 = 82 nM T02551 CCL54H 72187663 EC50 = 160 nM T02551 CMPS48 72190766 Ki = 22.9 nM T02551 C4E8TR 72191064 Ki = 110.7 nM T02551 C85FKU 72191065 Ki = 40.1 nM T02551 CNPA07 72191066 Ki = 2.7 nM T02551 CQL1T2 72191067 Ki = 132.5 nM T02551 CI2M7H 72191068 Ki = 134.6 nM T02551 C3ATN5 72197484 IC50 = 271.5 nM T02551 C20HSN 72197485 IC50 = 674.3 nM T02551 CN8A5R 72197486 IC50 = 807.3 nM T02551 CL3BF7 72197668 IC50 = 940.7 nM T02551 C7AOY4 72198754 IC50 = 24 nM T02551 C4M7KP 72198756 IC50 = 31 nM T02551 C0U5RS 72544566 Ki = 800 nM T02551 CVY4I0 72544787 Ki = 5700 nM T02551 C8UM5H 72544789 Ki = 1700 nM T02551 CVU61Z 72545007 Ki = 5100 nM T02551 CR6HY3 72545008 Ki = 7600 nM T02551 CC25RP 72545009 Ki = 17000 nM T02551 CW9OZ7 72545010 Ki = 25000 nM T02551 C14DJV 72545011 Ki = 17000 nM T02551 C4E5ZF 72545238 Ki = 2800 nM T02551 CY7J8U 72545239 Ki = 200 nM T02551 CU72QA 72545240 Ki = 2900 nM T02551 C4AS0E 72699528 Ki = 0.095 nM T02551 CO20CN 72699532 Ki = 0.058 nM T02551 C8EVJ6 72699690 Ki = 0.062 nM T02551 CEAK86 72699692 Ki = 0.4 nM T02551 CIR7G1 72699716 Ki = 19.93 nM T02551 COH4F8 72699779 Ki = 1.6 nM T02551 CIDS43 72699817 Ki = 39.86 nM T02551 C26STM 72700473 Ki = 0.16 nM T02551 CL96GC 72700475 Ki = 0.27 nM T02551 C45JKS 72700476 Ki = 0.19 nM T02551 C3TO8B 72700557 Ki = 0.047 nM T02551 CVA2X7 72700634 Ki = 0.09 nM T02551 CC01EJ 72737728 Ki = 2770 nM T02551 C6XYJ3 72737730 Ki = 2770 nM T02551 C6IF9H 72737744 Ki = 2770 nM T02551 CC65OA 73213195 Ki = 1496 nM T02551 CW83DK 73213196 Ki > 10000 nM T02551 CCV91B 73346042 Ki = 22 nM T02551 CK0HR9 73346334 Ki = 8662 nM T02551 C5QYH1 73347474 Ki = 1 nM T02551 CW8A0Y 73349359 Ki = 1048 nM T02551 C6BS5L 73349361 Ki > 10000 nM T02551 CY2IB5 73349362 Ki > 10000 nM T02551 C8GQK9 73350823 Ki = 6790 nM T02551 CV1U7L 73352414 Ki > 10000 nM T02551 CPZT87 73352849 Ki = 100 nM T02551 CCIT57 73353534 Ki = 4.3 nM T02551 C1NJ0R 73353884 Ki = 2685 nM T02551 C4F7VK 73355415 Ki = 5365 nM T02551 CX17VZ 73670899 IC50 = 6.8 nM T02551 CG21OC 73671061 Ki = 32 nM T02551 CS82XC 73671062 Ki = 36 nM T02551 CKW82D 73671216 IC50 = 0.4 nM T02551 CU5S6G 73671217 IC50 = 0.3 nM T02551 C7AJU1 73671218 IC50 = 0.3 nM T02551 CL4F9C 73671219 Ki = 20 nM T02551 CLS83G 73671367 Ki = 29 nM T02551 C2E7QW 75201901 Ki = 7900 nM T02551 C8IDL3 75306277 Ki = 31.62 nM T02551 CTH23U 76309672 Ki = 870.5 nM T02551 C08KCY 76309673 Ki = 14.7 nM T02551 C5OYN0 76311261 Ki = 0.43 nM T02551 C2VAS4 76311270 Ki = 1.5 nM T02551 CX40CG 76311272 Ki = 2 nM T02551 CZFW19 76314267 Ki = 23.99 nM T02551 C8QJ2B 76314861 Ki = 3.2 nM T02551 CIYJ90 76316875 Ki = 95.3 nM T02551 CQM65S 76318472 Ki = 3.8 nM T02551 CX9ON0 76318474 Ki = 0.9 nM T02551 CGZP35 76318476 Ki = 0.18 nM T02551 CD16XI 76320592 Ki = 56 nM T02551 CIB40D 76321554 Ki = 5.623 nM T02551 CS9F1X 76321556 Ki = 21.88 nM T02551 CJH2U5 76322139 Ki = 8.4 nM T02551 CG4EX6 76322141 Ki = 3 nM T02551 C97LOB 76325150 Ki = 2.884 nM T02551 CCR29U 76325152 Ki = 9.12 nM T02551 C6GBK1 76325154 Ki = 32.36 nM T02551 CLP59V 76325156 Ki = 19.05 nM T02551 C3K6UP 76325763 Ki = 4.4 nM T02551 C2O0FW 76328713 Ki = 1.66 nM T02551 C17YTI 76328715 Ki = 8.71 nM T02551 C97XIE 76329028 EC50 = 3.42 nM T02551 C0ED1J 76329346 Ki = 4 nM T02551 CHRD95 76331467 Ki = 35.4 nM T02551 CL2N3Y 76332978 Ki = 1.1 nM T02551 CC16RS 76332985 Ki = 3.1 nM T02551 CLJ16D 76332987 Ki = 3.7 nM T02551 CV1O9C 76332989 Ki = 0.39 nM T02551 CSW58A 76336021 Ki = 37.15 nM T02551 CL2I3A 76336596 Ki = 3.7 nM T02551 C1UZ5J 76441180 Ki = 2.1 nM T02551 C28RIZ 76518514 Ki = 9.7 nM T02551 CWI52H 77974401 Ki > 1000 nM T02551 CEAC35 85469680 EC50 = 0.912 nM T02551 C5JH2Y 85470564 EC50 = 0.302 nM T02551 C8EWX5 85658088 Ki = 324 nM T02551 CJ9N5Q 86280005 Ki = 0.351 nM T02551 CUA89I 86341962 Ki = 0.058 nM T02551 CWPH45 86341996 Ki = 0.043 nM T02551 CCR8X7 86342061 Ki = 0.055 nM T02551 CY2I8J 86342094 Ki = 1.2 nM T02551 CC47HJ 86342098 Ki = 0.18 nM T02551 CK03YC 86342156 Ki = 0.13 nM T02551 C5AQK2 86342192 Ki = 0.056 nM T02551 C9DZ2I 86342193 Ki = 0.31 nM T02551 CQP38R 86342194 Ki = 0.029 nM T02551 CE39OD 86342294 Ki = 0.043 nM T02551 CD7R6P 90213677 Ki = 9.6 nM T02551 CT8HK6 90389439 Ki = 424 nM T02551 CU9ED1 90389592 Ki = 480 nM T02551 CU8L2K 90466425 EC50 = 2.291 nM T02551 CVY5W3 90466571 EC50 = 2.1 nM T02551 CIM5O2 90466573 EC50 = 0.9 nM T02551 CFDK42 90466574 EC50 = 1 nM T02551 C1HQP6 90466717 EC50 = 2.6 nM T02551 CI1SR6 90466864 EC50 = 150 nM T02551 C5GX4U 90466867 EC50 = 19.95 nM T02551 C82YRS 90467020 EC50 = 6.9 nM T02551 C6B8ZY 90467021 EC50 = 15 nM T02551 C39ZDS 90467022 EC50 = 11 nM T02551 CT0N3V 90467024 EC50 = 1.4 nM T02551 CE8J9X 90467168 EC50 = 3.6 nM T02551 CTQG73 90467169 EC50 = 240 nM T02551 C76CLR 90467172 EC50 = 120 nM T02551 C7T0BR 90467173 EC50 = 130 nM T02551 C8JXQ1 90467317 EC50 = 1200 nM T02551 CF3QC2 90467318 EC50 = 14 nM T02551 CG34EY 90467320 EC50 = 330 nM T02551 CB61FX 90467322 EC50 = 12 nM T02551 C8C1KA 90467323 EC50 = 3.9 nM T02551 CYB97T 90467452 EC50 = 37 nM T02551 CYUQ73 90467453 EC50 = 4 nM T02551 C2WVX1 90467587 EC50 = 4.4 nM T02551 CB6I7A 90643699 Ki = 37.9 nM T02551 C3EY5T 90643700 Ki = 22.1 nM T02551 CKYP81 90643701 Ki = 2.61 nM T02551 CF5U1L 90643702 Ki = 2.8 nM T02551 C80SXV 90644057 Ki = 354.81 nM T02551 C20EPB 90644058 Ki = 2477 nM T02551 C04MRN 90644059 Ki = 4534 nM T02551 CIA8J4 90644060 Ki = 2772 nM T02551 CY8TP0 90644061 Ki = 187 nM T02551 CKV24H 90644062 Ki = 158.49 nM T02551 CW2ZC4 90644063 Ki = 156 nM T02551 CLG60I 90644064 Ki = 119 nM T02551 CKLN72 90644065 Ki = 180 nM T02551 C7G5VH 90644066 Ki = 2290 nM T02551 CLM0J5 90644067 Ki = 1340 nM T02551 CQL6N2 90644068 Ki = 33 nM T02551 CQ7OJ1 90644069 Ki = 850 nM T02551 CGY80L 90644070 Ki = 670.7 nM T02551 CDPE48 90644071 Ki = 1462 nM T02551 CLFV10 90644226 Ki = 2.1 nM T02551 CZ7LD8 90644227 Ki = 1.3 nM T02551 C35GPQ 90644228 EC50 = 5 nM T02551 CZI30L 90644230 Ki = 1.9 nM T02551 CUO0J6 90644928 Ki = 6.9 nM T02551 CF9HI4 90644929 Ki = 29 nM T02551 CX2WE7 90644930 Ki = 560 nM T02551 C4MUI2 90664601 IC50 = 493 nM T02551 CHT7D5 90664962 IC50 = 2189 nM T02551 CACG19 90666899 Ki = 1348.96 nM T02551 CODM50 90666903 Ki = 1096.48 nM T02551 C0J5YH 91864602 Ki = 16.98 nM T02551 CUQ6V0 92042918 Ki < 1000 nM T02551 C3S6VX 92209551 IC50 = 1.6 nM T02551 CCV0I4 92640710 Ki = 25900 nM T02551 COA3U6 102262219 Ki = 1700 nM T02551 CE6Z3M 109030343 Ki = 781 nM T02551 CC1P6O 109030515 Ki = 4530 nM T02551 CTYH92 117028759 Ki > 39319 nM T02551 C7P5RX 117869686 Ki = 253 nM T02551 C59ZAJ 117870140 Ki = 12 nM T02551 CS8YG9 117870408 Ki = 19 nM T02551 CJ7KU8 117870413 Ki = 524 nM T02551 C95QKZ 117870490 Ki = 9.3 nM T02551 CU5S8B 117870714 Ki = 134 nM T02551 CNM0U7 117870915 Ki = 99 nM T02551 CV80LK 117870976 Ki = 45 nM T02551 C5I4TZ 117871054 Ki = 8.4 nM T02551 C5HR9I 117871069 IC50 = 7.2 nM T02551 C1KDN4 117871083 Ki = 78 nM T02551 C2I0HB 118643968 Ki = 652 nM T02551 CJS6B2 118709159 Ki = 14 nM T02551 C9XDM6 118709160 Ki = 31 nM T02551 CQ9C5S 118709161 Ki = 11 nM T02551 C1YRW4 118709162 Ki = 11 nM T02551 CPL69Z 118709163 Ki = 6.4 nM T02551 CGAB49 118709164 Ki = 9.1 nM T02551 C3SX4Z 118709165 Ki = 39 nM T02551 CC7FW6 118709166 Ki = 210 nM T02551 CRMK67 118709167 Ki = 160 nM T02551 CW4YS6 118709168 Ki = 220 nM T02551 CY3BR2 118709169 Ki = 380 nM T02551 CIX72C 118709170 Ki = 82 nM T02551 C2O8BG 118709171 Ki = 500 nM T02551 COV8K7 118709172 Ki = 270 nM T02551 CJZD82 118709173 Ki = 9.5 nM T02551 C16WQU 118709174 Ki = 47 nM T02551 C4E5MK 118709175 Ki = 30 nM T02551 CFV2M0 118709176 Ki = 1.8 nM T02551 C08TAX 118709177 Ki = 5.9 nM T02551 CYNM75 118709178 Ki = 9.8 nM T02551 CJZ7G0 118709179 Ki = 19 nM T02551 CSB25E 118709750 Ki = 11 nM T02551 CD4S9R 118709751 Ki = 1.3 nM T02551 CBG0D4 118710458 Ki = 10 nM T02551 CR90MQ 118710459 IC50 = 0.0038 nM T02551 CN9HD5 118710460 IC50 = 1.8 nM T02551 C13SFN 118710461 Ki = 6.4 nM T02551 CIWT51 118710462 Ki = 124 nM T02551 CZ2HV3 118710463 Ki = 77 nM T02551 CW1I6Z 118710464 Ki = 2014 nM T02551 CW14NI 118710465 Ki = 148 nM T02551 CZ7WQ3 118710466 IC50 = 5.6 nM T02551 CK2XE7 118710467 Ki = 4.3 nM T02551 CFBT50 118710468 Ki = 32 nM T02551 CR97VN 118710469 Ki = 35 nM T02551 C9CJ5R 118710470 IC50 = 14 nM T02551 CZSB43 118710935 Ki = 745 nM T02551 CX6NP5 118710936 Ki = 1141 nM T02551 CB5VH9 118710937 Ki = 1100 nM T02551 CDJZ51 118710938 Ki = 64 nM T02551 CQ5Z8V 118710939 Ki = 512 nM T02551 CWGD39 118710940 Ki = 120 nM T02551 CL8SA7 118710941 Ki = 512 nM T02551 CEY68Q 118710942 Ki = 575 nM T02551 CM8P2H 118710943 Ki = 279 nM T02551 CHL2U8 118710944 Ki = 502 nM T02551 CVHK79 118710945 Ki = 477 nM T02551 CG8PJ0 118710947 Ki = 115 nM T02551 C3GW0U 118710948 Ki = 73 nM T02551 C9QB7F 118710949 Ki = 129 nM T02551 CMJ0S5 118710950 Ki = 144 nM T02551 CO8E9F 118711252 Ki > 1000 nM T02551 CJY9D7 118711253 Ki > 1000 nM T02551 CFJE45 118711254 Ki > 1000 nM T02551 CM47VI 118711261 Ki > 1000 nM T02551 CX3M2Z 118711262 Ki > 1000 nM T02551 C4UAV9 118711266 Ki > 1000 nM T02551 C83MBF 118711267 Ki > 1000 nM T02551 C9FH2L 118711268 Ki > 1000 nM T02551 C4R3NA 118714496 Ki = 0.75 nM T02551 C8AUL2 118714497 Ki = 0.62 nM T02551 CW8F2K 118714498 Ki = 0.67 nM T02551 CE89TI 118714552 Ki = 2770 nM T02551 CE5M8O 118719791 Ki = 22.2 nM T02551 C8M1VO 118719792 Ki = 4.7 nM T02551 CQY62K 118719793 Ki = 3.1 nM T02551 C97UXN 118719794 Ki = 36.3 nM T02551 CG0O3Q 118719795 Ki = 3.7 nM T02551 CUHT71 118719796 Ki = 1.8 nM T02551 CR0FM7 118719797 Ki = 8.9 nM T02551 CPX2Y1 118719798 Ki = 8.2 nM T02551 C0KH8S 118719799 Ki = 6.3 nM T02551 C4YR6K 118719800 Ki = 26.5 nM T02551 CX7WL5 118719801 Ki = 6.5 nM T02551 C5TO1H 118719802 Ki = 3.2 nM T02551 CTQ71B 118719803 Ki = 93.1 nM T02551 C8KJ6Y 118719804 Ki = 25.4 nM T02551 CFL6U9 118719805 Ki = 21.1 nM T02551 CQK7O2 118719806 Ki = 29.6 nM T02551 CWO13F 118719807 Ki = 13.9 nM T02551 CZ8FE6 118719808 Ki = 6.7 nM T02551 CRH56E 118719809 Ki = 9.6 nM T02551 CUH0A6 118719810 Ki = 2.3 nM T02551 CZKW38 118719811 Ki = 6.8 nM T02551 C74DCE 118719812 Ki = 2.9 nM T02551 CT8KO4 118719925 Ki = 588.84 nM T02551 C16DHZ 118719926 Ki = 676.08 nM T02551 CLA06I 118719927 Ki = 954.99 nM T02551 CYW82N 118721287 Ki > 1000 nM T02551 CES97Y 118722639 Ki = 0.3 nM T02551 CM3P7R 118722912 Ki = 204 nM T02551 CP3QC2 118722913 Ki = 3 nM T02551 C1PG3C 118722914 Ki = 16 nM T02551 CR6E5D 118722915 Ki = 24 nM T02551 CTE58Z 118730369 Ki = 500 nM T02551 COS3K9 121304408 Ki = 0.1585 nM T02551 C9G3ZJ 121304414 Ki = 0.8511 nM T02551 CVN57T 121304417 Ki = 2.089 nM T02551 C4RD9Y 121304424 Ki = 6.166 nM T02551 CN5YP1 121304426 Ki = 0.2089 nM T02551 CJ4GF7 121304428 Ki = 15.14 nM T02551 CXL97W 121304430 Ki = 1.995 nM T02551 CA8CY5 121304437 Ki = 0.2754 nM T02551 C1PKR0 121304441 Ki = 0.4677 nM T02551 CQ7T4P 121304448 Ki = 3.236 nM T02551 CWLB20 121304449 Ki = 2.399 nM T02551 CC3MP6 121304452 Ki = 0.06761 nM T02551 CW68KD 121304458 Ki = 5.495 nM T02551 CVA9F4 121304464 Ki = 1.445 nM T02551 CPB58L 121304467 Ki = 1.738 nM T02551 CFXN81 121304470 Ki = 3.236 nM T02551 CTCA98 121304474 Ki = 1.445 nM T02551 COB2X5 121304477 Ki = 3.311 nM T02551 CZ0BI4 121304484 Ki = 36.31 nM T02551 CW51NQ 121304485 Ki = 0.631 nM T02551 CX1DQ6 121304488 Ki = 7.079 nM T02551 CZ4D2Y 121304493 Ki = 3.631 nM T02551 CU50JM 121304499 Ki = 1.259 nM T02551 C7NLV2 121304500 Ki = 1.479 nM T02551 C18GSY 121304506 Ki = 41.69 nM T02551 C21MEQ 121304510 Ki = 0.263 nM T02551 C7F3NO 121304514 Ki = 1.047 nM T02551 CPNV43 121304527 Ki = 0.3311 nM T02551 CCW3A9 121304532 Ki = 1.82 nM T02551 CQ2UM4 121304538 Ki = 0.3388 nM T02551 CR7L0O 121304539 Ki = 0.5495 nM T02551 C2GI6S 121304542 Ki = 3.311 nM T02551 C1AB6P 121304551 Ki = 0.5248 nM T02551 CTI6Z7 121304565 Ki = 2.57 nM T02551 CFVP28 121304568 Ki = 1.38 nM T02551 CO6JN7 121304569 Ki = 0.182 nM T02551 CN05ZQ 121304574 Ki = 4.074 nM T02551 CU0M7B 121304590 Ki = 3.981 nM T02551 C3FPD2 121304592 Ki = 89.13 nM T02551 C73GOE 121304594 Ki = 25.12 nM T02551 CLZK90 121304596 Ki = 3.981 nM T02551 C6YLM8 121304597 Ki = 1.288 nM T02551 CX5MO3 121304598 Ki = 2.754 nM T02551 C12GJP 121304609 Ki = 6.761 nM T02551 C6DT8C 121304616 Ki = 25.12 nM T02551 CZS7C4 121304618 Ki = 75.86 nM T02551 CDQ35E 121304633 Ki = 28.84 nM T02551 C31AEQ 121304649 Ki = 0.4169 nM T02551 C9TYS1 121304653 Ki = 1.995 nM T02551 C2VTK5 121304654 Ki = 0.6761 nM T02551 CQY2T8 121304655 Ki = 128.82 nM T02551 CSYD40 121304673 Ki = 27.54 nM T02551 C6IB0P 121304685 Ki = 8.71 nM T02551 CU0L6A 121304697 Ki = 17.78 nM T02551 CNOW27 121304705 Ki = 1.738 nM T02551 C6NA0P 121304710 Ki = 2.692 nM T02551 CXC70Q 121304711 Ki = 1.175 nM T02551 CE0ND7 121304744 Ki = 0.3162 nM T02551 C1MZ6T 121304754 Ki = 10 nM T02551 CU93LN 121304777 Ki = 19.95 nM T02551 C5HQ4S 121304867 Ki = 1.047 nM T02551 CAS0Y9 121315197 Ki = 21.38 nM T02551 CG92LO 121315203 Ki = 5.129 nM T02551 CRZ1V0 121315205 Ki = 0.9772 nM T02551 CV3XH6 121315206 Ki = 1.514 nM T02551 C4TI7P 121315244 Ki = 0.7943 nM T02551 CLM9E8 121315259 Ki = 53.7 nM T02551 C7B3XN 121315293 Ki = 25.12 nM T02551 C9U5CV 121315295 Ki = 22.39 nM T02551 C6UMN2 121315304 Ki = 26.3 nM T02551 CH5FS4 121315329 Ki = 97.72 nM T02551 CX71KH 121315331 Ki = 29.51 nM T02551 CV4EO5 121315336 Ki = 1.38 nM T02551 CN39AK 121315339 Ki = 1.096 nM T02551 CFWG90 121315351 Ki = 10 nM T02551 C14NCL 121315356 Ki = 1.023 nM T02551 COG90M 121315374 Ki = 1.66 nM T02551 CEY62R 121315401 Ki = 0.537 nM T02551 C0NB3Y 121315426 Ki = 16.6 nM T02551 C0E6HD 121315586 Ki = 0.4169 nM T02551 CA7HL6 121315615 Ki = 19.95 nM T02551 CBAG84 121315634 Ki = 0.5754 nM T02551 C35WTP 122177641 Ki = 0.63 nM T02551 C8OS7B 122177642 Ki = 2.2 nM T02551 CV2AT4 122177644 Ki = 1.2 nM T02551 CB16GY 122177645 Ki = 0.21 nM T02551 CP6VX4 122180568 Ki = 2.93 nM T02551 CU0L3S 122180569 Ki = 1.59 nM T02551 C87MAH 122180570 Ki = 3.1 nM T02551 CY9BN0 122180571 Ki = 13.1 nM T02551 CS9NY8 122180572 Ki = 3.8 nM T02551 CAL57I 122180573 Ki = 5.05 nM T02551 CZ72GE 122180574 Ki = 1 nM T02551 CZ4M2F 122180575 Ki = 11.1 nM T02551 C03CGT 122180576 Ki = 5.55 nM T02551 C2X3ZW 122180610 Ki = 5.48 nM T02551 CRMS80 122180611 Ki = 6.73 nM T02551 CWO2Y4 122180612 Ki = 5.88 nM T02551 C2DZ0K 122180613 Ki = 7.7 nM T02551 CH81IV 122180614 Ki = 14 nM T02551 C1EPB8 122180615 Ki = 1.47 nM T02551 CV26IM 122180616 Ki = 1.35 nM T02551 CQ0L6Z 122180617 Ki = 8.32 nM T02551 CVX5Y3 122180618 Ki = 40.7 nM T02551 CEGV53 122180619 Ki = 30.5 nM T02551 CV1OA4 122180620 Ki = 173 nM T02551 CYID81 122180621 Ki = 493 nM T02551 CB91ZG 122180622 Ki = 18.5 nM T02551 C1CIH2 122180623 Ki = 68.2 nM T02551 C8YZ9Q 122180624 Ki = 25.2 nM T02551 C9S3VH 122180625 Ki = 55.8 nM T02551 CQ3N6G 122180626 Ki = 33.6 nM T02551 C6YL5S 122180627 Ki = 5.85 nM T02551 CPRB82 122180954 Ki = 1.4 nM T02551 C08BVN 122180955 Ki = 2.8 nM T02551 CH9SX5 122180956 Ki = 87 nM T02551 CAJ9N8 122181005 Ki = 18 nM T02551 C90VEH 122181006 Ki = 2.91 nM T02551 CN7TP8 122181007 Ki = 0.233 nM T02551 CCV9D5 122181326 Ki = 3 nM T02551 C91LDR 122181327 Ki = 0.72 nM T02551 CPW19F 122181328 Ki = 1.4 nM T02551 C5D1NC 122181329 Ki = 0.31 nM T02551 C05RGV 122181330 Ki = 0.85 nM T02551 C1KWI9 122181331 Ki = 2 nM T02551 CQ35XD 122181332 Ki = 4.9 nM T02551 C3XGN0 122181333 Ki = 14 nM T02551 C3BTQ7 122181334 Ki = 2.11 nM T02551 CXL5V3 122183764 Ki = 3.63 nM T02551 CK3VT8 122183765 Ki = 1.99 nM T02551 CQ6CW2 122183766 Ki = 31.6 nM T02551 CQE64Y 122183767 Ki = 0.57 nM T02551 CI43NJ 122183768 Ki = 8.05 nM T02551 CK6D3O 122183769 Ki = 0.392 nM T02551 CC2WO0 122183770 Ki = 0.907 nM T02551 C12TRH 122183771 Ki = 0.118 nM T02551 CZO5G4 122183772 Ki = 0.173 nM T02551 C8V5TM 122183773 Ki = 0.244 nM T02551 CH4J7G 122183774 Ki = 0.128 nM T02551 CKIP60 122183775 Ki = 97.9 nM T02551 C8AK5V 122183776 Ki = 2.51 nM T02551 CS65WU 122183777 Ki = 53.1 nM T02551 C06GQO 122183778 EC50 = 0.95 nM T02551 C8YL2R 122183779 Ki = 2.14 nM T02551 CQ4YF9 122183780 Ki = 44.8 nM T02551 C7ZNJ8 122183781 Ki = 52.9 nM T02551 C4U8LC 122183782 Ki = 69.9 nM T02551 CLA65S 122183783 Ki = 37.7 nM T02551 CIG04A 122186385 Ki = 87.6 nM T02551 C6UI5G 122186390 Ki = 3.9 nM T02551 C6LN7X 122186408 Ki = 9.4 nM T02551 C4FUN7 122187390 Ki = 570.88 nM T02551 CI7F8R 122187393 Ki = 1140.65 nM T02551 C25WZN 122188153 Ki = 43 nM T02551 CE0VY6 122188155 Ki = 15.7 nM T02551 CY6O8L 122188157 Ki = 3.3 nM T02551 CURK46 122188159 Ki = 9.9 nM T02551 CK5BP3 122189387 Ki = 77 nM T02551 C8JV3W 122189388 Ki = 12 nM T02551 CV1U4Q 122189389 Ki = 4.4 nM T02551 C4PBA3 122189390 Ki = 32 nM T02551 CD7UN3 122189391 Ki = 8.5 nM T02551 C14FCX 122189392 Ki = 2.2 nM T02551 C1NIK8 122189393 Ki = 8.5 nM T02551 C9KXH4 122189394 Ki = 0.31 nM T02551 C87LIY 122191600 Ki = 18000 nM T02551 CPF1G4 122191601 Ki = 2300 nM T02551 C3ZR7F 122191602 Ki = 1300 nM T02551 CI5L4E 122191603 Ki = 600 nM T02551 C9AH4E 122191604 Ki = 620 nM T02551 CVJ3R4 122191605 Ki = 200 nM T02551 CSR76G 122191606 Ki = 280 nM T02551 C2J4ZX 122191607 Ki = 89 nM T02551 CM84TD 122191608 Ki = 4300 nM T02551 C94XIT 122191609 Ki = 1800 nM T02551 C7UVD4 122191610 Ki = 4600 nM T02551 CWH1P8 122191611 Ki = 930 nM T02551 C7ODW3 122195524 Ki > 900 nM T02551 C71KZQ 122205437 Ki = 24 nM T02551 C30ZRC 122205438 Ki = 18 nM T02551 C6TEJ0 126532768 Ki = 5.012 nM T02551 CNRI41 126533424 Ki = 3.981 nM T02551 CG65RM 126533453 Ki = 12.59 nM T02551 CRX67M 126533461 Ki = 1.995 nM T02551 C0OPY6 126533669 Ki = 0.3162 nM T02551 CSN21X 126533798 Ki = 1.995 nM T02551 CMHY08 126533799 Ki = 3.981 nM T02551 CP8W0X 126533801 Ki = 7.943 nM T02551 CXM45K 126533810 Ki = 0.1995 nM T02551 C0E7OY 126533847 Ki = 10 nM T02551 CPL62Z 126533872 Ki = 0.7943 nM T02551 C1ST0Y 126533877 Ki = 7.943 nM T02551 CDP5C4 126533939 Ki = 3.162 nM T02551 CX2A4N 126533957 Ki = 2.512 nM T02551 CIV7R0 126533969 Ki = 6.31 nM T02551 CC7V5Y 126533978 Ki = 1 nM T02551 CI97TU 126533981 Ki = 1.585 nM T02551 CON63X 126534012 Ki = 3.162 nM T02551 C9G1IV 126534022 Ki = 0.1995 nM T02551 C9AN4B 126534041 Ki = 1.585 nM T02551 C8JKG0 126534069 Ki = 3.162 nM T02551 C65OJB 126534075 Ki = 39.81 nM T02551 CA4QM3 126534084 Ki = 2.512 nM T02551 C3SUR8 126534086 Ki = 5.012 nM T02551 CCX0O5 126534178 Ki = 7.943 nM T02551 C6NU0Y 126534182 Ki = 12.59 nM T02551 CNUA81 126534195 Ki = 1.259 nM T02551 CIAD86 126534204 Ki = 7.943 nM T02551 C4R7XU 126534291 Ki = 3.981 nM T02551 CVBX50 126534373 Ki = 1.259 nM T02551 CB94HO 126534441 Ki = 7.943 nM T02551 CSX9W5 126534443 Ki = 31.62 nM T02551 CQ39ZD 126534462 Ki = 6.31 nM T02551 CT75WF 126534466 Ki = 5.012 nM T02551 C52IHK 126534498 Ki = 3.162 nM T02551 CFA3D6 126534516 Ki = 0.7943 nM T02551 CX14VB 126534676 Ki = 0.631 nM T02551 CIW18V 126534678 Ki = 0.3162 nM T02551 CGA1E9 126534722 Ki = 31.62 nM T02551 CJPA49 126534738 Ki = 1.995 nM T02551 CG7CY3 126534740 Ki = 0.1995 nM T02551 CQDE96 126534746 Ki = 15.85 nM T02551 CIN62J 126534758 Ki = 1.585 nM T02551 CXI58O 126534764 Ki = 50.12 nM T02551 C0WUJ5 126534771 Ki = 1.259 nM T02551 CFDR90 126534824 Ki = 50.12 nM T02551 CX9LM7 126534859 Ki = 3.981 nM T02551 CKN57U 126534860 Ki = 1.995 nM T02551 C3YB2Z 126534863 Ki = 2.512 nM T02551 CR70LT 126534933 Ki = 2.512 nM T02551 CKBT37 126534948 Ki = 5.012 nM T02551 C6DLR7 126534986 Ki = 3.981 nM T02551 CR10PO 126534991 Ki = 25.12 nM T02551 CFT24J 126535001 Ki = 1.995 nM T02551 C58EIM 126535029 Ki = 12.59 nM T02551 C5HQB6 126535034 Ki = 0.3981 nM T02551 C9Q0VB 126535075 Ki = 5.012 nM T02551 CMT3Q8 126535410 Ki = 12.59 nM T02551 C95HVE 126535414 Ki = 12.59 nM T02551 C5YS6F 126535470 Ki = 1 nM T02551 C4TZ6I 126535517 Ki = 12.59 nM T02551 CM57GR 126720252 Ki = 1600 nM T02551 CCF0J2 127024958 Ki = 12.7 nM T02551 C82TLX 127024959 Ki = 1.23 nM T02551 C2MWE6 127024960 Ki = 10.4 nM T02551 C9AQH0 127025258 Ki = 1.33 nM T02551 CH1CG6 127025275 Ki = 3.9 nM T02551 CG3N7S 127025276 Ki = 1.3 nM T02551 CGO8I5 127025277 Ki = 1.8 nM T02551 CJZC96 127025278 Ki = 2 nM T02551 CQ60XE 127025279 Ki = 123 nM T02551 CTBN56 127026052 Ki = 120.23 nM T02551 CG8Q4L 127026123 Ki = 0.73 nM T02551 C2YDB4 127027076 Ki = 1.1 nM T02551 CU59DP 127027077 Ki = 0.2 nM T02551 CI94GN 127027078 Ki = 1.3 nM T02551 C2H6GE 127027079 Ki = 0.5 nM T02551 C5G4AH 127027080 Ki = 3.5 nM T02551 C9PNV3 127027384 Ki = 1.6 nM T02551 C09YOS 127027905 Ki > 10000 nM T02551 CH2BP0 127027974 Ki = 12 nM T02551 CXQ94C 127028034 Ki = 87 nM T02551 CE9MN1 127028185 Ki > 10000 nM T02551 C8MC1I 127028408 Ki = 194.98 nM T02551 C9SC6E 127028505 Ki > 10000 nM T02551 C1RF0I 127031156 Ki = 125.89 nM T02551 CJ4YC0 127031397 Ki = 101 nM T02551 CBU9G2 127031398 Ki = 220 nM T02551 CE1IA7 127031399 Ki = 110 nM T02551 C4WKG9 127031403 Ki = 54 nM T02551 CEDM28 127031404 Ki = 1367 nM T02551 CV5UH0 127031405 Ki = 1811 nM T02551 CHN9X2 127031422 Ki = 44 nM T02551 C0CY9W 127031423 Ki = 53 nM T02551 CNH2V8 127031424 Ki = 65 nM T02551 C0A3PY 127031458 Ki = 125.89 nM T02551 C2W0HL 127031949 Ki = 2680 nM T02551 CQ0ZT9 127035062 Ki = 498 nM T02551 CO53TS 127035828 Ki > 1000 nM T02551 CY7LP9 127035829 Ki > 1000 nM T02551 CR29BS 127035830 Ki > 1000 nM T02551 CU49VE 127036186 Ki = 691.83 nM T02551 CG06BD 127036932 Ki = 141.25 nM T02551 CVW71O 127036953 Ki = 239.88 nM T02551 CT1Z3P 127037852 Ki > 10000 nM T02551 CH6KI9 127037866 Ki > 10000 nM T02551 C81TYN 127038069 Ki = 810 nM T02551 C0SWK3 127038076 Ki = 290 nM T02551 C3QL9U 127038078 Ki = 270 nM T02551 CP8T3I 127039208 Ki > 10000 nM T02551 CBF6T8 127039745 EC50 = 1.41 nM T02551 CLY0X5 127039746 EC50 = 3.93 nM T02551 CAW01Z 127040356 Ki = 12.59 nM T02551 CZ6V5D 127040357 Ki > 10000 nM T02551 CE95PL 127040381 Ki > 10000 nM T02551 C37KDY 127040382 Ki = 10 nM T02551 C6Z9VL 127040695 Ki = 15.85 nM T02551 CQGJ12 127040696 Ki = 19.95 nM T02551 CWC31L 127040697 Ki > 10000 nM T02551 CF31EG 127040698 Ki > 10000 nM T02551 CMH9E6 127040712 Ki > 10000 nM T02551 CG74QA 127040713 Ki = 15.85 nM T02551 CZ58KA 127040714 Ki > 10000 nM T02551 C34BGK 127040715 Ki = 6.31 nM T02551 CL4WG3 127040716 Ki > 10000 nM T02551 C53WRO 127041026 Ki = 19.95 nM T02551 C0S5MT 127041332 Ki > 10000 nM T02551 C5B1AG 127041347 Ki = 39.81 nM T02551 C0J8HC 127041348 Ki = 3.162 nM T02551 C8MG6H 127041349 Ki > 10000 nM T02551 C87MZF 127041350 Ki > 10000 nM T02551 CT5LX7 127041672 Ki > 10000 nM T02551 C9D7SK 127041673 Ki > 10000 nM T02551 CS78AZ 127041951 Ki > 10000 nM T02551 CU9C4S 127041952 Ki = 25.12 nM T02551 C9HPT6 127041953 Ki = 15.85 nM T02551 C4FG7S 127042371 EC50 = 10.9 nM T02551 C7ETU0 127042372 EC50 = 0.84 nM T02551 CM02RK 127045814 EC50 = 53.7 nM T02551 C35GAL 127045853 Ki = 690 nM T02551 C17LBT 127045854 Ki = 400 nM T02551 CJ8GS7 127045855 Ki = 2200 nM T02551 CZN72J 127046238 EC50 = 20.6 nM T02551 CT15OK 127046255 Ki = 21.7 nM T02551 C1CR3G 127046595 EC50 = 7.4 nM T02551 C3WNA8 127046749 Ki = 27200 nM T02551 C59QDV 127046922 EC50 = 53 nM T02551 C2E1ZA 127046948 Ki = 790 nM T02551 CTI5Z8 127046949 Ki = 18 nM T02551 C4D6BQ 127046950 Ki = 62 nM T02551 CM4CQ7 127046951 Ki = 660 nM T02551 C29ERQ 127046952 Ki = 12 nM T02551 C9DFA6 127047182 EC50 = 21.7 nM T02551 C78IFA 127047221 Ki = 610 nM T02551 CFOD25 127047227 Ki = 10.3 nM T02551 C5CG1O 127047229 Ki = 3.39 nM T02551 CN3B7M 127047230 EC50 = 19.6 nM T02551 CD24JH 127047310 EC50 = 14.4 nM T02551 C9FQ0O 127047316 EC50 = 11.2 nM T02551 C28FLN 127047317 EC50 = 6.6 nM T02551 CU2ST0 127047318 EC50 = 6.8 nM T02551 C6TMB2 127047319 EC50 = 6.3 nM T02551 CB80KL 127047458 EC50 = 10.5 nM T02551 C81BCP 127047461 EC50 = 76.5 nM T02551 C1D7PX 127047462 EC50 = 14.1 nM T02551 C0RE8Z 127047592 EC50 = 19.2 nM T02551 C4S3IQ 127047593 EC50 = 57.8 nM T02551 C9J7QI 127047594 EC50 = 37.7 nM T02551 CI64SZ 127047595 EC50 = 25.4 nM T02551 CTZ3W9 127047639 EC50 = 11.4 nM T02551 C71MFW 127047640 EC50 = 6.9 nM T02551 C6P4OZ 127047641 EC50 = 7.5 nM T02551 CZL0U7 127047859 Ki = 3.5 nM T02551 C4SG7L 127047870 EC50 = 30.7 nM T02551 CZ6XL5 127047996 Ki = 25 nM T02551 C3G8BQ 127048020 EC50 = 11.9 nM T02551 CC7BU0 127049059 Ki = 20.89 nM T02551 C42FHY 127049060 Ki = 31 nM T02551 CF2QY9 127049061 Ki = 162.18 nM T02551 CX53AC 127050632 Ki = 499 nM T02551 CTL0S1 127051516 Ki = 32 nM T02551 CTL8J1 127051843 Ki = 336 nM T02551 CF6V9Q 127051844 Ki = 13 nM T02551 C8TNB1 127051845 Ki = 38 nM T02551 CT9O7G 127051863 Ki = 942 nM T02551 C5ONG1 127051864 Ki = 12.88 nM T02551 CVQW26 127051865 Ki = 16 nM T02551 CRF85X 127052458 Ki = 143 nM T02551 CCY71I 127052465 Ki = 630 nM T02551 C2E9VX 127052467 Ki = 467.74 nM T02551 CPO4C3 127052468 Ki = 162 nM T02551 CSQ2N8 127052486 Ki = 109 nM T02551 C4YJ8H 127052487 Ki = 50.12 nM T02551 CT9RS4 127052488 Ki = 31.62 nM T02551 CLU7C1 127052757 Ki = 6007 nM T02551 C95KYT 127052758 Ki = 769 nM T02551 CYNR02 127052759 Ki = 117.49 nM T02551 C14YJU 127052778 Ki = 233 nM T02551 C1JAS7 127052779 Ki = 28 nM T02551 C7MQK8 127053042 Ki = 161 nM T02551 C3WIA6 129103318 IC50 = 25.6 nM T02551 C10VDB 130431277 EC50 = 17.9 nM T02551 CI1NF8 130431279 Ki = 446 nM T02551 CS8O4E 130431287 Ki = 3.19 nM T02551 C75AQS 130431288 Ki = 0.84 nM T02551 C85MOW 130431289 Ki = 0.756 nM T02551 CR7T6X 130431290 Ki = 1.14 nM T02551 C2OH7B 130431291 Ki = 99.9 nM T02551 C2AZ0H 130431294 Ki = 13 nM T02551 CEQ43Y 130431295 Ki = 27.9 nM T02551 CK64GU 130431296 Ki = 2.45 nM T02551 CU9XL0 130431303 Ki = 11.2 nM T02551 CB6Q3Y 130431306 Ki = 35.3 nM T02551 C3MA6H 130431309 Ki = 4.23 nM T02551 CYW0X2 130431314 Ki = 0.29 nM T02551 C8ZED9 130431315 Ki = 0.373 nM T02551 CDN26V 130431316 Ki = 0.362 nM T02551 CL64UW 130431317 Ki = 0.985 nM T02551 C8HE2O 130431318 Ki = 6.84 nM T02551 CZ6S4T 130431319 Ki = 0.886 nM T02551 C8ZHI7 130431325 Ki = 0.153 nM T02551 CF5SW8 130431328 Ki = 37.9 nM T02551 CN9RZ3 130431329 Ki = 7.4 nM T02551 CEP1Q6 130431334 Ki = 0.2 nM T02551 CWT8I6 130431336 Ki = 1.28 nM T02551 CN70MW 130431337 Ki = 0.142 nM T02551 CIXV41 130431340 Ki = 0.621 nM T02551 C4GF1U 130431342 Ki = 36.1 nM T02551 CWAC20 130431343 Ki = 0.331 nM T02551 C2WI5R 130431351 Ki = 0.341 nM T02551 C50GOC 130442480 Ki = 8100 nM T02551 CM04RF 130442572 Ki > 10000 nM T02551 CLP6B7 130816094 Ki = 424 nM T02551 C7FM0U 132060763 Ki = 264 nM T02551 CT81OY 132060776 Ki = 951 nM T02551 CFXL21 132060812 Ki = 175 nM T02551 C3HI8S 132141090 Ki = 12.3 nM T02551 CU5F7W 132141173 Ki = 10.72 nM T02551 C5P9AV 132153537 Ki = 7.943 nM T02551 C3CVU2 132156264 Ki = 35.48 nM T02551 C9W4AK 132156266 Ki = 15.14 nM T02551 CRH07J 132156331 Ki = 2.754 nM T02551 CF5V3G 132156412 Ki = 7.762 nM T02551 CCL8F6 132495282 Ki = 398.11 nM T02551 CR7TA8 132495283 Ki = 1258.93 nM T02551 CVZ57M 132578416 EC50 = 0.33 nM T02551 CAVB41 132584404 Ki > 10000 nM T02551 CY4CU6 132606870 Ki = 0.89 nM T02551 CVYX78 132606872 Ki = 32 nM T02551 C6Z5UG 134129927 Ki = 1000 nM T02551 C8O2EP 134130246 Ki = 79.43 nM T02551 CLW62U 134131970 Ki = 501.19 nM T02551 C7UOA9 134132432 Ki > 10000 nM T02551 CQX4U3 134133064 Ki > 10000 nM T02551 CCPI30 134133464 Ki = 1.4 nM T02551 C0J2ML 134133604 Ki = 776.25 nM T02551 CP0E5M 134133632 Ki = 150 nM T02551 CM0TS6 134133967 Ki = 30.2 nM T02551 CR8HL3 134134147 Ki = 4.571 nM T02551 CR4F6X 134135492 Ki = 0.052 nM T02551 CM34TY 134135507 Ki = 0.31 nM T02551 CJ6C3E 134135947 Ki > 10000 nM T02551 CGX03A 134136246 Ki = 88 nM T02551 CFOU70 134136921 Ki = 1995.26 nM T02551 C87ZJW 134137152 Ki > 10000 nM T02551 CSM98N 134137323 Ki = 2070 nM T02551 CD41CW 134137432 Ki = 0.046 nM T02551 C50WSG 134137966 Ki = 1258.93 nM T02551 C90XZH 134138881 Ki = 0.051 nM T02551 C2DK7E 134139144 Ki = 125.89 nM T02551 CTP83K 134139510 Ki = 0.22 nM T02551 C5RTN3 134139606 Ki = 373 nM T02551 CLW86T 134141354 Ki = 338.84 nM T02551 CXC80B 134142146 Ki = 8.7 nM T02551 CVJ70S 134143778 Ki = 0.21 nM T02551 CJE86B 134143833 Ki = 175 nM T02551 CL8I1U 134144243 Ki = 19.95 nM T02551 CR5L4K 134144303 Ki = 106 nM T02551 C0J1IR 134145434 Ki = 726 nM T02551 C8AZ1F 134146083 Ki = 1.1 nM T02551 C8RI0E 134146106 Ki = 7.3 nM T02551 CC9P2T 134146194 Ki = 524.81 nM T02551 CZDH24 134147097 Ki = 251.19 nM T02551 CV4WJ5 134147644 Ki = 630.96 nM T02551 CB0NS6 134147903 Ki = 3213 nM T02551 CH21YW 134148634 Ki = 3162.28 nM T02551 CJ5W4V 134149077 Ki = 450 nM T02551 CBU81N 134149168 Ki > 10000 nM T02551 CUFG17 134150400 Ki = 195 nM T02551 CSE17M 134150535 Ki = 251.19 nM T02551 C0S2VH 134150637 Ki = 2.63 nM T02551 C5DX6R 134150645 Ki = 3171 nM T02551 C6NYU2 134150754 Ki = 2.188 nM T02551 C2MAK7 134150852 Ki = 3605 nM T02551 C6O8QW 134150900 Ki = 1258.93 nM T02551 CLU34D 134151427 Ki = 866 nM T02551 CW7AH9 134151737 Ki = 131 nM T02551 C8BI7V 134151764 Ki = 195 nM T02551 CK23XB 134151891 Ki = 0.14 nM T02551 CNC39L 134151926 Ki = 1258.93 nM T02551 CB16CR 134152436 Ki = 1584.89 nM T02551 CI0G7H 134153418 Ki = 0.24 nM T02551 CB6M5Y 134153538 Ki = 91 nM T02551 C42ZDI 134153624 Ki = 1000 nM T02551 C79TEI 134154068 Ki = 446.68 nM T02551 C9DQ4Y 134154208 Ki = 0.78 nM T02551 CMJ1U3 134154387 Ki = 184 nM T02551 C4VGJ5 134154679 Ki = 1071.52 nM T02551 CU6C4G 134154943 Ki = 1 nM T02551 C6QAY2 134155116 Ki = 223 nM T02551 CM6D4G 134155367 Ki = 1258.93 nM T02551 C79QLN 134155460 Ki = 2176 nM T02551 CW5VZ9 134155502 Ki = 106 nM T02551 C0AE1P 134156091 Ki = 794.33 nM T02551 CVR87Q 134156222 Ki = 66 nM T02551 C08MHZ 134157446 Ki = 31 nM T02551 C4DZ5M 135418440 Ki > 7900 nM T02551 CZXW36 135469096 Ki > 7900 nM T02551 C8XYU4 135481864 Ki = 3437 nM T02551 C1MTS9 135492584 Ki = 1811 nM T02551 C7RQ2Y 135506137 Ki > 7900 nM T02551 C0TY5Z 135514603 IC50 = 52 nM T02551 C2U1EP 135524323 Ki = 960 nM T02551 CH96LU 135559170 Ki = 2200 nM T02551 CNQ47X 135846033 Ki = 1.259 nM T02551 CG95BM 135887931 Ki > 4000 nM T02551 CQYI85 135887934 Ki = 408 nM T02551 C5W7CT 135887940 Ki > 1000 nM T02551 C5KE3N 135986088 Ki = 223 nM T02551 CJEK87 135995891 Ki = 7600 nM T02551 C89VLZ 136056636 Ki = 0.86 nM T02551 CZR53O 136072267 Ki = 167 nM T02551 CKJY95 137040409 Ki = 3.981 nM T02551 CA9L5S 137631807 Ki = 83.9 nM T02551 C1VMC5 137631956 Ki = 256 nM T02551 C5QI2K 137632035 Ki = 115 nM T02551 C3LDV7 137632586 Ki = 390 nM T02551 CN8BJ2 137632607 Ki = 3.7 nM T02551 C3R2LO 137632761 Ki = 2.7 nM T02551 C3PF9Z 137633454 Ki = 3.2 nM T02551 CSA30N 137633662 Ki = 2.47 nM T02551 COF9I6 137633705 Ki = 2.2 nM T02551 C8YM6U 137633863 EC50 = 0.32 nM T02551 CN1I7A 137634153 Ki = 110 nM T02551 C8EG5N 137634366 EC50 = 3.7 nM T02551 C6FRJ5 137634397 Ki = 0.35 nM T02551 CM54XV 137635157 Ki = 94.2 nM T02551 CPHI76 137635364 Ki = 0.31 nM T02551 C8ZFQ6 137635685 Ki = 50 nM T02551 C6QB9W 137635734 Ki = 3981.07 nM T02551 CGEQ16 137635743 Ki = 373 nM T02551 CZ36LE 137636066 Ki = 2 nM T02551 CIV34M 137636185 Ki = 1090 nM T02551 CAL1W4 137636298 Ki = 1700 nM T02551 CX8O0V 137636308 Ki = 3890.45 nM T02551 CAQ6I5 137636351 Ki = 1.7 nM T02551 C6GWQ3 137636460 EC50 = 66 nM T02551 CQ20FO 137636498 Ki = 27 nM T02551 CZU6N5 137636581 Ki = 200 nM T02551 C0YDQ5 137637428 Ki = 790 nM T02551 C8U7ZW 137637481 Ki = 377 nM T02551 CF7KG5 137637817 Ki = 19.6 nM T02551 CXO70S 137638203 Ki = 139 nM T02551 CPQ98N 137638817 Ki = 690 nM T02551 C49VDK 137638973 Ki = 0.41 nM T02551 CA03VC 137639125 Ki = 66.07 nM T02551 C1HX3Z 137639304 Ki = 510 nM T02551 C51HEL 137639330 Ki = 119 nM T02551 CC16HE 137640152 Ki = 1.6 nM T02551 CZP68A 137640189 Ki = 1 nM T02551 CZ4TA9 137640201 Ki = 1819.7 nM T02551 CB2NO0 137640203 Ki = 7.4 nM T02551 CV49MZ 137640371 Ki = 1.6 nM T02551 CN4ST6 137640376 Ki = 235 nM T02551 CCU7L3 137640391 Ki = 28 nM T02551 C1EK3W 137640451 Ki = 25.6 nM T02551 CX4A3N 137640511 Ki = 3715.35 nM T02551 C8IO0R 137640836 Ki = 8.5 nM T02551 C6PU4A 137640863 EC50 = 3.7 nM T02551 CI1TU3 137641550 Ki = 141 nM T02551 CWXF83 137641643 Ki = 192 nM T02551 C6PT7L 137642033 Ki = 5.9 nM T02551 C94WSH 137642380 Ki = 5.6 nM T02551 C4Q6ZM 137642607 Ki = 707.95 nM T02551 CPX85V 137642676 Ki = 34.7 nM T02551 CUT21E 137642921 Ki = 140 nM T02551 CAC6W0 137643122 Ki = 30 nM T02551 C71XIQ 137643132 Ki = 1.2 nM T02551 CK51LB 137643309 Ki = 1.1 nM T02551 C3O0FX 137643951 Ki = 70 nM T02551 C0HS3L 137644131 Ki = 1040 nM T02551 C34PUI 137644833 Ki = 7.4 nM T02551 C0KL6Q 137644962 Ki = 2630.27 nM T02551 CVX6T1 137644966 Ki = 2.3 nM T02551 C4PV8U 137645196 Ki = 42 nM T02551 CPCY48 137645406 Ki = 12 nM T02551 CNH95X 137645574 Ki = 12 nM T02551 C3TP2G 137645830 Ki = 40 nM T02551 C2L4CG 137645834 Ki = 1.51 nM T02551 CG8P6I 137645938 Ki = 281.84 nM T02551 C96EAP 137646245 Ki = 33.88 nM T02551 CPI68E 137646281 Ki = 6 nM T02551 C8C7UI 137647058 Ki = 558 nM T02551 C1C3YT 137647150 Ki = 4.12 nM T02551 CYH5U9 137647533 Ki = 240 nM T02551 CWY02V 137648255 Ki = 75.2 nM T02551 C5XL4K 137648359 Ki = 600 nM T02551 C0X4WB 137649193 Ki = 4790 nM T02551 CH9WS3 137649435 Ki = 0.31 nM T02551 CVYC51 137649540 Ki = 833 nM T02551 C75ELQ 137649585 Ki = 2.45 nM T02551 C3IF6W 137649770 Ki = 1350 nM T02551 CFBL16 137650746 Ki = 0.45 nM T02551 C7BOY5 137650793 Ki = 2.8 nM T02551 C6R3IG 137650900 Ki = 438 nM T02551 CR3Z6M 137651073 Ki = 12 nM T02551 CW4T6D 137651322 Ki = 1.2 nM T02551 CS3OV1 137651866 Ki = 24.2 nM T02551 C15YDU 137651936 EC50 = 0.4266 nM T02551 CC9F7J 137652174 EC50 = 18 nM T02551 CS61YC 137652312 Ki = 871 nM T02551 C94NAQ 137652404 Ki = 23.4 nM T02551 CU8E4M 137652517 Ki = 113 nM T02551 C65RCN 137653034 Ki = 0.69 nM T02551 CX30HQ 137653096 Ki = 2800 nM T02551 C5ZJN8 137653359 Ki = 640 nM T02551 C32FLB 137653517 Ki = 0.172 nM T02551 CQ93DX 137653577 Ki = 2682 nM T02551 C48VDP 137653978 Ki = 80.6 nM T02551 C4C6EV 137653986 Ki = 160 nM T02551 COTX19 137654511 Ki = 380 nM T02551 CF5Y2A 137654675 Ki = 3.8 nM T02551 CLI4D8 137655029 Ki = 24 nM T02551 C7RW9H 137655451 Ki = 13 nM T02551 CJAZ13 137655556 Ki = 3.4 nM T02551 C6CA5H 137655594 Ki = 420 nM T02551 CUC54G 137655636 Ki = 407.38 nM T02551 CDAN02 137655735 Ki = 13 nM T02551 CD16SQ 137655795 Ki = 38 nM T02551 CMA0T6 137655799 Ki = 169 nM T02551 CI68MV 137655953 Ki = 382 nM T02551 CLT53E 137656298 Ki = 34.3 nM T02551 CJO23S 137656836 Ki = 51.7 nM T02551 CA7F5N 137657115 Ki = 3.2 nM T02551 CV2CR4 137657153 Ki = 11 nM T02551 C1HA0D 137657276 Ki = 23.4 nM T02551 CE0Y7P 137657322 Ki = 2.3 nM T02551 CRT86S 137657427 Ki = 1.9 nM T02551 CH76FP 137657951 Ki = 48 nM T02551 CY4H6C 137658100 EC50 = 17 nM T02551 C5F8AB 137658819 Ki = 0.5 nM T02551 CEZ07P 137659303 Ki = 15 nM T02551 CT9YA5 137659335 Ki = 97.7 nM T02551 CG2U9R 137659809 Ki = 210 nM T02551 CP9AN6 137659990 Ki = 0.59 nM T02551 CP6US4 137660046 Ki = 0.71 nM T02551 CF0KP5 137660062 EC50 = 1.2 nM T02551 C8W3AQ 137660395 Ki = 77.7 nM T02551 CKIH14 137660417 EC50 = 1.66 nM T02551 C5V4DQ 137660707 Ki = 7.7 nM T02551 C1VB2N 137660751 Ki = 598 nM T02551 C42IDE 137660837 EC50 = 0.4786 nM T02551 CG8QR9 137660855 Ki = 9.81 nM T02551 CDA8V2 137661377 Ki = 1548.82 nM T02551 C5X9LH 137661635 EC50 = 0.9 nM T02551 CZI74G 137661939 Ki = 82.4 nM T02551 CT3P2B 137662048 Ki = 181888 nM T02551 C9YXI5 137662136 Ki = 227 nM T02551 C7WJT2 142573371 Ki = 101 nM T02551 CT3SY0 142573376 Ki = 2773 nM T02551 C9B0JX 142573379 Ki = 75 nM T02551 CQO6K2 142573380 Ki = 59.2 nM T02551 CEXL42 142573384 Ki = 33.3 nM T02551 CJIC89 142573385 Ki = 32.5 nM T02551 CAL25K 142573386 Ki = 138 nM T02551 C5BOX1 142573395 Ki = 45.1 nM T02551 CX6S8U 142573399 Ki = 57 nM T02551 CIZ75U 142573404 Ki = 48.7 nM T02551 CXI8C3 142573405 Ki = 61.5 nM T02551 CG2H3O 142573406 Ki = 112 nM T02551 C1L0GO 142573412 Ki = 63 nM T02551 CCY49O 142573415 Ki = 213 nM T02551 CFX0W5 142573417 Ki = 1098 nM T02551 C09XCG 142573420 Ki = 208 nM T02551 C1IBV7 142573422 Ki = 25.4 nM T02551 CQ0E4W 142573428 Ki = 92.9 nM T02551 CB5M2G 142573431 Ki = 3.2 nM T02551 CNZX48 142573438 Ki = 370 nM T02551 CQ5W7B 142573439 Ki = 6647 nM T02551 C7G3NO 142573444 Ki = 383 nM T02551 CN5WK4 142573449 Ki = 89.7 nM T02551 CK42UE 142592111 Ki = 160 nM T02551 CM03WS 142592130 Ki = 505 nM T02551 CL58XS 145967572 Ki = 19 nM T02551 C58WSL 145967904 Ki = 162 nM T02551 CB1FD8 145968810 Ki = 13.49 nM T02551 C48XNG 145969667 Ki = 2.344 nM T02551 CNZY06 145969934 Ki = 49 nM T02551 C61MSO 145970938 Ki = 131 nM T02551 C1XF0I 145979855 Ki = 22 nM T02551 CO12QR 145979897 Ki = 10 nM T02551 C87MSW 145980271 Ki = 782 nM T02551 CW5TE2 145980543 Ki = 410 nM T02551 C3N5DH 145981580 Ki = 28 nM T02551 CP6DT9 145986441 Ki = 3.4 nM T02551 CNJH37 145986752 Ki = 437 nM T02551 CO4LK7 145988180 Ki = 41 nM T02551 C0RY8X 145988474 Ki = 6.3 nM T02551 CUGO10 145988693 Ki = 474 nM T02551 C4P6IC 145989012 Ki = 5.9 nM T02551 CBN7D9 145990000 EC50 = 0.026 nM T02551 CLF26V 145990141 Ki = 2.1 nM T02551 C6NYE9 145990254 EC50 = 1.1 nM T02551 CPW28Y 145990453 Ki = 2.7 nM T02551 CW87TZ 145991769 Ki = 12 nM T02551 CCP2U1 145992489 Ki = 552 nM T02551 C74MRE 145993220 Ki = 24 nM T02551 CRWE54 145993377 Ki = 2.7 nM T02551 CT29LQ 145993700 Ki = 8.7 nM T02551 C4TY6L 145993896 EC50 = 0.00048 nM T02551 C2H5AO 145993990 Ki = 4.4 nM T02551 CC2G1V 146025727 Ki = 6200 nM T02551 CO9A5N 146451658 Ki = 3.02 nM T02551 C12RYJ 146451661 Ki = 23.6 nM T02551 C9MCB1 146451664 Ki = 4.31 nM T02551 C65FZJ 146451691 Ki = 24.5 nM T02551 C5ZOJ3 146680920 Ki = 150 nM T02551 CD1CB9 151199471 Ki = 133 nM T02551 CU9FD3 151880864 Ki = 23256 nM T02551 C6P3SR 153287553 Ki > 10000 nM T02551 CV9G7Z 153287572 Ki > 10000 nM T02551 CO85KL 153287574 Ki > 10000 nM T02551 CA9S3Y 155195287 Ki = 2130 nM T02551 C7XIR5 155195305 Ki = 26200 nM T02551 CQ5WA9 155195311 Ki = 1.85 nM T02551 CCFR96 155195429 Ki = 354 nM T02551 C3S2EX 155195430 Ki = 613 nM T02551 C0RQT6 155195433 Ki = 1590 nM T02551 CL61UG 155195435 Ki = 8660 nM T02551 C10GRK 155195439 Ki = 1150 nM T02551 CME84G 155195441 Ki = 1190 nM T02551 CQ3G0P 155195442 Ki = 73000 nM T02551 CH4BL7 155195444 Ki = 6470 nM T02551 C1JQ7Y 155195448 Ki = 6010 nM T02551 CM9RP4 155195449 Ki = 276 nM T02551 CON51V 155195451 Ki = 806 nM T02551 CL9Z5V 155195452 Ki = 31.2 nM T02551 CLQ72J 155195454 Ki = 1330 nM T02551 CUH20V 155195486 Ki = 282 nM T02551 CG5NW0 155195487 Ki = 34 nM T02551 CJK6C0 155195495 Ki = 21100 nM T02551 C6ZV8B 155195496 Ki = 5.96 nM T02551 CF3EY0 155195497 Ki = 11300 nM T02551 COJL79 155195501 Ki = 173 nM T02551 CD2EV4 155195516 Ki = 24200 nM T02551 C3MC0Q 155510756 Ki = 76 nM T02551 C13IEH 155511416 Ki = 3801.89 nM T02551 CTW28Q 155511803 Ki = 26320 nM T02551 CJ96WB 155512259 Ki = 88 nM T02551 C1YB7P 155512384 Ki = 12302.69 nM T02551 CQ83KZ 155512662 Ki = 0.5 nM T02551 C2TRB6 155512841 Ki = 14.7 nM T02551 C0DKF9 155512851 Ki = 3.8 nM T02551 C6XST7 155513053 Ki = 496 nM T02551 C6FEW4 155513265 Ki = 2378 nM T02551 C35GHL 155513375 Ki = 21.9 nM T02551 CD4Y8Z 155513529 Ki = 3090.3 nM T02551 C0ZXT4 155513773 Ki = 130 nM T02551 CHXY56 155513802 Ki = 26.7 nM T02551 CL5G9Q 155513837 Ki = 2.2 nM T02551 CX7A3L 155513965 Ki = 28.18 nM T02551 CF6K8R 155514137 Ki = 1400 nM T02551 CK9YN0 155514430 Ki = 22.5 nM T02551 CH34RK 155514798 Ki = 64.6 nM T02551 CV8F7A 155515301 Ki = 2884.03 nM T02551 C3XZM2 155515759 Ki = 320 nM T02551 CUE5J3 155515907 Ki = 4 nM T02551 CM65NQ 155515931 Ki = 160 nM T02551 CAS50P 155515966 Ki = 32.7 nM T02551 CUM2N4 155515982 Ki = 170 nM T02551 CV12SD 155516041 Ki = 1.5 nM T02551 CJ98ZK 155516236 Ki = 87.1 nM T02551 CH7N0C 155516494 Ki > 50000 nM T02551 CQY58Z 155516873 Ki = 2000 nM T02551 C9ZAW0 155517266 Ki = 43 nM T02551 C47LRQ 155518026 Ki = 220 nM T02551 C79MXU 155518617 Ki = 8.3 nM T02551 CPER92 155519378 Ki = 76 nM T02551 C0KLD8 155519559 Ki = 32 nM T02551 CUSA24 155519891 Ki > 10000 nM T02551 C8IYD1 155520455 Ki = 113.1 nM T02551 C5DSE0 155520996 Ki = 55 nM T02551 C7SG3T 155521675 Ki = 239.88 nM T02551 C9R5AM 155521711 Ki = 0.55 nM T02551 C5NM0F 155522454 EC50 = 0.78 nM T02551 CV7IG5 155522663 Ki = 104.7 nM T02551 CD59RE 155522719 Ki > 50000 nM T02551 C2H3JL 155523073 Ki = 15 nM T02551 CQA76T 155523112 Ki = 11.1 nM T02551 C3E9DJ 155523127 Ki = 45.4 nM T02551 CG6Y4Z 155523515 Ki = 110 nM T02551 CVQ68Y 155523770 Ki = 14.5 nM T02551 COH1Q5 155524191 Ki = 4.4 nM T02551 CW7NT8 155524423 Ki = 2.6 nM T02551 CQX27T 155525357 Ki = 39.4 nM T02551 CT0NV4 155525431 Ki > 50000 nM T02551 CT1YQ0 155525527 EC50 = 2.62 nM T02551 CW65KS 155525705 Ki = 26.9 nM T02551 CPZ0H7 155526424 Ki = 16.7 nM T02551 C9ANR8 155527358 Ki = 21 nM T02551 C9IW8F 155527714 Ki = 120 nM T02551 CGA2J9 155528048 Ki = 446.68 nM T02551 CU69ZH 155529400 Ki = 3.02 nM T02551 CEN90X 155529453 Ki = 614 nM T02551 CUSG17 155529568 Ki = 120 nM T02551 C8U7QC 155529592 Ki = 85 nM T02551 CBS2O8 155529683 Ki > 30000 nM T02551 C8WC5Y 155530733 Ki = 700 nM T02551 CDGX72 155530763 Ki = 510 nM T02551 CCGZ20 155530937 Ki > 10000 nM T02551 C95JRV 155531663 EC50 = 1.22 nM T02551 C4VK0L 155531809 Ki = 1800 nM T02551 C3R4YM 155532148 Ki = 257.04 nM T02551 CKZ35G 155532475 Ki = 106.3 nM T02551 C4LOR5 155532477 Ki = 549.6 nM T02551 CK9JP0 155532505 Ki = 92 nM T02551 CZA89B 155533824 Ki = 13.6 nM T02551 CQ12KS 155533996 Ki = 32.6 nM T02551 C8AX5N 155534186 Ki = 23.4 nM T02551 CZTX89 155534246 Ki = 130 nM T02551 CC4D5K 155535057 Ki = 2.42 nM T02551 C71YMQ 155535169 Ki = 104.71 nM T02551 CGZ5T8 155535272 Ki = 0.363 nM T02551 C3V1CL 155535404 Ki = 1145 nM T02551 CA3N2X 155535680 Ki = 3801.89 nM T02551 CHP2Z9 155535866 Ki = 25.7 nM T02551 CA01QX 155536022 Ki = 860 nM T02551 CB79ZW 155536080 Ki > 10000 nM T02551 CDL9R5 155536374 Ki = 104.71 nM T02551 CDEX60 155536720 Ki = 1246 nM T02551 CY61EO 155536815 Ki = 3681 nM T02551 CFCG03 155537361 Ki = 61 nM T02551 C6NT4F 155537490 Ki = 257.04 nM T02551 CVFD68 155537516 EC50 = 3.58 nM T02551 C13CSU 155537907 Ki = 23.7 nM T02551 CP3WK6 155538028 Ki = 660 nM T02551 C2S9LF 155538235 Ki = 27.8 nM T02551 CFPT03 155538349 Ki = 1500 nM T02551 C75SRB 155538429 Ki = 1.5 nM T02551 C3DIY2 155539246 Ki = 89.8 nM T02551 CAOV97 155539413 Ki = 418 nM T02551 CPV48W 155539557 Ki = 84.5 nM T02551 CBT04Y 155539651 Ki = 208 nM T02551 CJD9C8 155540541 Ki = 173 nM T02551 C8WRH2 155540919 Ki = 75.86 nM T02551 C58YSH 155542160 Ki = 525 nM T02551 CM9FI1 155542182 Ki = 640 nM T02551 C7U3JN 155542198 Ki = 24 nM T02551 CC51DL 155542687 Ki = 78.3 nM T02551 CVK2M9 155543189 Ki = 15.5 nM T02551 CDO05U 155543223 Ki = 449 nM T02551 C3UXC2 155543605 EC50 = 3500 nM T02551 C4ANI0 155543691 Ki = 5.3 nM T02551 CIEQ43 155543869 Ki = 72 nM T02551 C08FTE 155544239 Ki = 1.2 nM T02551 CJBP49 155546194 Ki = 401 nM T02551 C7MCZ0 155546478 Ki = 11.2 nM T02551 C9D0GL 155547128 Ki = 140 nM T02551 C1SVX6 155547259 Ki = 173 nM T02551 CA9K1Y 155547729 Ki = 25.9 nM T02551 CUGC98 155547873 Ki = 0.89 nM T02551 CECV12 155548038 Ki = 39.8 nM T02551 CM4XB6 155548127 Ki = 27 nM T02551 CJ7AL8 155548205 Ki = 26 nM T02551 C9GM0D 155548336 Ki = 1800 nM T02551 C54AQR 155549026 Ki = 1672 nM T02551 C0DHX7 155550192 Ki = 19 nM T02551 CU93YK 155550351 Ki = 330 nM T02551 CN6I4P 155550431 Ki = 45.7 nM T02551 C3Y1EJ 155550445 Ki = 13.6 nM T02551 CY34NR 155550580 Ki = 73 nM T02551 C6N9PG 155550640 Ki = 55.8 nM T02551 CG7NR9 155550756 Ki = 26.5 nM T02551 CHXB35 155551102 Ki = 212 nM T02551 C82QWR 155551173 Ki = 23.4 nM T02551 CX8JA1 155552185 Ki = 310 nM T02551 CY94BV 155552356 Ki = 108 nM T02551 CMS62Z 155552380 Ki = 95 nM T02551 CG70XQ 155552591 Ki = 17.6 nM T02551 CB4F8Y 155552676 Ki = 524.8 nM T02551 C0DQ3Z 155552695 Ki = 179 nM T02551 CV9SY1 155552989 Ki = 688 nM T02551 CP6KN4 155553364 Ki = 36.1 nM T02551 C1RLI0 155553370 Ki > 10000 nM T02551 C6STK4 155553745 Ki = 383 nM T02551 CN3Z2Q 155553911 Ki = 19.8 nM T02551 CD5LC6 155554006 Ki = 11.5 nM T02551 CCA21K 155554569 Ki = 562 nM T02551 CELU08 155555060 Ki = 150 nM T02551 CLN79H 155555200 Ki = 362 nM T02551 CWY29E 155555201 Ki = 40.9 nM T02551 C1RCM0 155555224 Ki = 16 nM T02551 C5Q4UP 155555402 Ki = 517 nM T02551 C76IMR 155555589 Ki = 33.88 nM T02551 C1I5JR 155556665 Ki = 631 nM T02551 CQ6YT5 155557645 Ki = 14587 nM T02551 C3UCM2 155557792 Ki = 537.03 nM T02551 CE7MX4 155557986 Ki = 103 nM T02551 C36SYJ 155558844 Ki = 23.4 nM T02551 CGBZ63 155559617 Ki = 25 nM T02551 C06BZW 155559811 Ki = 48 nM T02551 C1U4ZL 155560181 Ki = 147.91 nM T02551 C60GZE 155560295 Ki = 1900 nM T02551 CD61BM 155560516 Ki = 0.2 nM T02551 C7OZM6 155561446 Ki = 20.8 nM T02551 C75RMN 155561496 Ki = 3 nM T02551 CD2L9R 155561779 Ki = 280 nM T02551 CALB48 155561861 Ki = 0.44 nM T02551 CTZE48 155561895 Ki = 309.03 nM T02551 CF89GP 155562328 Ki = 86 nM T02551 C2Z0HB 155562353 Ki = 562.3 nM T02551 CRMC43 155562395 Ki > 10000 nM T02551 C2EBQ1 155562463 Ki = 165.96 nM T02551 CH0PW5 155562681 Ki = 18 nM T02551 CV4PM8 155562984 Ki = 0.25 nM T02551 C4IH5Z 155563301 Ki > 10000 nM T02551 C1KU5D 155563347 Ki = 25.7 nM T02551 C5KCZ1 155563589 EC50 = 20.4 nM T02551 CAZL19 155563950 Ki = 1300 nM T02551 CU7JG9 155564308 Ki = 95 nM T02551 C54WIE 155564667 Ki = 0.941 nM T02551 C0UN4V 155564747 Ki = 31.6 nM T02551 C2QLX9 155565138 Ki = 121 nM T02551 CIB3R0 155565292 Ki = 17 nM T02551 C4OZ2X 155565438 Ki = 0.47 nM T02551 CMH8I1 155565768 Ki = 33.1 nM T02551 CYIG07 155566058 Ki = 400 nM T02551 C0Y9RV 155566355 Ki = 0.68 nM T02551 CRJG23 155566403 Ki = 1100 nM T02551 CK20WA 155566662 Ki = 36.7 nM T02551 C7P8GE 155566829 Ki = 712 nM T02551 CEV3B9 155566852 Ki = 68 nM T02551 CN12ES 155566888 Ki = 227 nM T02551 C6DPR8 155566974 Ki = 12.8 nM T02551 C46ZDJ 155567045 Ki = 8 nM T02551 CCR6S2 155567442 Ki = 321 nM T02551 C6I5QA 155567666 Ki = 591 nM T02551 C4NX7P 155567775 Ki = 0.41 nM T02551 C95RAP 155567835 Ki = 218.8 nM T02551 C5A6YM 155567869 Ki = 2 nM T02551 C8NO4X 155567971 Ki = 850 nM T02551 CRX8J2 155568278 Ki = 194.98 nM T02551 CQ5N6X 155568411 Ki > 50000 nM T02551 C7FR1Q 155568415 Ki = 72753 nM T02551 CHO2G1 155568612 Ki = 396 nM T02551 CVU42Z 155568628 Ki = 5.7 nM T02551 CV24CW 155568676 Ki = 18.8 nM T02551 C73ERT 155568786 Ki = 44 nM T02551 CKG5M1 155568867 EC50 = 2802 nM T02551 C42JKO 155569198 Ki = 3.8 nM T02551 C3N9VU 10251906 Ki > 500 nM T02551 CP9TR0 10324985 Ki = 62.8 nM T02551 C9J5HY 16105548 Ki = 0.37 nM T02551 C4ZD3A 16105549 Ki = 0.45 nM T02551 CFMK68 3246545 Ki = 23 nM T02551 D00CDM 115107 Ki > 10000 nM T02551 D00HUV 9881815 Ki = 67.2 nM T02551 D00NQV 5041 Ki = 145 nM T02551 D00SDJ 11237664 Ki = 0.8 nM T02551 D01ENR 2993172 Ki > 10000 nM T02551 D01JXM 46222048 Ki > 1000 nM T02551 D01KIH 44323762 Ki = 870.5 nM T02551 D01WWC 16573 Ki > 950 nM T02551 D02NNS 9845181 Ki = 59 nM T02551 D02YDU 10420539 Ki = 13000 nM T02551 D03DET 10287730 Ki = 1000 nM T02551 D03GES 9995378 Ki = 6800 nM T02551 D03JOS 233952 Ki = 280 nM T02551 D03JOX 11311147 IC50 > 10000 nM T02551 D03KUH 57267 Ki = 0.11 nM T02551 D03PYX 1219 EC50 = 0.531 nM T02551 D04AZE 3277600 Ki < 31622.78 nM T02551 D04CPW 25139331 Ki = 11000 nM T02551 D04CTN 11074524 Ki = 52 nM T02551 D04PBA 10015867 Ki = 28.9 nM T02551 D04RBU 45486362 Ki = 0.57 nM T02551 D04TWX 9794475 EC50 = 8 nM T02551 D05BCJ 2779264 Ki = 15000 nM T02551 D05EQG 5265 Ki = 0.12 nM T02551 D05HMW 10705550 Ki = 1600 nM T02551 D05NQX 9961911 Ki = 10 nM T02551 D05QJK 9816808 Ki = 8.8 nM T02551 D05XGR 6918647 Ki = 794.33 nM T02551 D05ZUX 44207909 Ki >= 1000 nM T02551 D06AIQ 107995 Ki = 4.2 nM T02551 D06FUV 5311189 EC50 = 9.8 nM T02551 D06HTJ 24866612 EC50 = 0.085 nM T02551 D06LQH 167715 Ki = 0.44 nM T02551 D06NTB 30438 Ki = 6700 nM T02551 D06QGD 11357862 IC50 > 10000 nM T02551 D06VDN 443391 IC50 > 1000 nM T02551 D06WLB 9838216 Ki = 19.5 nM T02551 D07GQP 11477180 Ki = 0.316 nM T02551 D07LRJ 5312149 Ki = 501.19 nM T02551 D07RYR 44396235 Ki = 1818 nM T02551 D07UUQ 15508240 Ki = 7900 nM T02551 D07VBS 10425450 Ki = 167 nM T02551 D07ZOP 11470616 IC50 > 10000 nM T02551 D08CKM 9863250 Ki = 1258.93 nM T02551 D08TCX 11437461 Ki = 4654 nM T02551 D09CFW 57377246 Ki = 4100 nM T02551 D09CVG 449126 Ki > 4400 nM T02551 D09FTZ 10564794 Ki = 3500 nM T02551 D09PIN 3378093 Ki > 1000 nM T02551 D09PJF 44588498 Ki = 1.77 nM T02551 D09RPR 16737207 Ki > 10000 nM T02551 D09WBJ 10336538 Ki = 46 nM T02551 D0A2BE 2780 Ki = 10.4 nM T02551 D0AX0K 5615 IC50 = 5500 nM T02551 D0B9DR 15508243 Ki = 2600 nM T02551 D0C0UM 10775317 Ki = 13000 nM T02551 D0D1PR 130907 Ki = 1.02 nM T02551 D0E1PL 9865384 Ki = 10000 nM T02551 D0E1RX 11335419 Ki = 2923 nM T02551 D0E3AL 56597938 Ki = 1.9 nM T02551 D0F0IA 11301655 Ki > 6000 nM T02551 D0F6CD 5202 EC50 = 523 nM T02551 D0FF6S 16038374 IC50 > 10000 nM T02551 D0FU2V 24754478 Ki = 0.825 nM T02551 D0G2CP 10404144 Ki = 3890.45 nM T02551 D0G8CV 9954003 Ki = 0.5012 nM T02551 D0G8VU 3645619 Ki = 2810 nM T02551 D0H2WQ 54562 EC50 = 0.097 nM T02551 D0H3KU 172267 EC50 = 0.14 nM T02551 D0H3WJ 44435193 Ki = 8900 nM T02551 D0H7PC 6918553 Ki > 5011.87 nM T02551 D0H9QG 5312148 Ki = 3981.07 nM T02551 D0I9KV 11220599 IC50 > 10000 nM T02551 D0IU8V 9903877 Ki = 2.8 nM T02551 D0J1HP 10378389 Ki = 2.4 nM T02551 D0K3UL 9796720 Ki = 560 nM T02551 D0L5MW 181743 Ki = 309 nM T02551 D0L7OM 6917970 Ki = 30 nM T02551 D0LV7U 10667433 Ki = 195 nM T02551 D0M2BB 25333445 Ki = 2100 nM T02551 D0M2ZE 6604756 Ki = 4 nM T02551 D0M3PV 133633 Ki = 48.6 nM T02551 D0M5XV 24866114 EC50 = 0.06 nM T02551 D0M7SY 9910352 Ki = 1.995 nM T02551 D0M8LN 9806160 Ki = 1.3 nM T02551 D0NA2T 24800688 Ki = 130 nM T02551 D0O1PM 4420454 EC50 = 4.4 nM T02551 D0O3GF 1220 Ki = 259 nM T02551 D0O4BC 11776546 Ki = 11 nM T02551 D0O7DA 37459 Ki = 0.04 nM T02551 D0O9BZ 2728532 Ki = 35.4 nM T02551 D0OG0R 10337743 IC50 > 5000 nM T02551 D0P0IX 16104 IC50 = 120 nM T02551 D0PN9R 16655023 Ki = 375 nM T02551 D0PV6G 115007 Ki = 12.59 nM T02551 D0Q4DP 6603897 Ki > 4500 nM T02551 D0Q5IP 10851078 Ki = 95 nM T02551 D0Q7FM 15443 Ki = 53 nM T02551 D0R3GW 10296414 Ki = 630.96 nM T02551 D0R5QM 10354670 Ki = 23.9 nM T02551 D0R8UU 44396220 Ki = 7804 nM T02551 D0S1XN 44323962 Ki = 56 nM T02551 D0S7WZ 5119 Ki = 249 nM T02551 D0SL4Q 46190878 Ki > 10000 nM T02551 D0T1TU 68950 Ki = 4667 nM T02551 D0T2RY 9948320 Ki >= 1000 nM T02551 D0T3IH 119146 Ki = 0.265 nM T02551 D0TU5W 44323978 Ki = 95.3 nM T02551 D0V4NW 25139332 Ki = 950 nM T02551 D0V4RP 1346 Ki = 2262 nM T02551 D0W1HM 3408722 Ki = 0.11 nM T02551 D0WD6J 10357869 Ki = 770 nM T02551 D0WU9R 133008 Ki = 480 nM T02551 D0X1QW 122334 Ki = 26 nM T02551 D0X8LG 11243002 IC50 > 10000 nM T02551 D0Y8UC 3929516 Ki = 145 nM T51452 D07JVL 3016 Ki = 17 nM T51452 D0L9GG 2118 EC50 = 12 nM T51452 D0T1WN 5732 EC50 = 737 nM T51452 D0CH7C 57336276 Ki = 502 nM T51452 D0HO2T 23581869 Ki = 0.3 nM T51452 D0Z9HW 23630026 Ki = 5 nM T51452 C1Z6YU 9821389 Ki = 26 nM T51452 CCX58U 9865233 Ki = 2 nM T51452 C7BA0Z 9908880 Ki = 0.7 nM T51452 C1VRB9 9951530 EC50 = 101 nM T51452 CPC3U1 9971547 Ki = 180 nM T51452 CUT5W8 9976743 EC50 = 99 nM T51452 CUSM85 10221761 Ki = 0.6 nM T51452 CFBW42 10883539 Ki = 0.3 nM T51452 CBQ4R7 10905261 EC50 = 188 nM T51452 C15NXT 10926766 EC50 = 1179 nM T51452 CK1S7J 10927005 EC50 = 67 nM T51452 CWK02D 10936672 EC50 = 1162 nM T51452 C09PCZ 10971225 EC50 = 210 nM T51452 CG9Z6N 10991911 EC50 = 184 nM T51452 C7DVK8 11014215 EC50 = 154 nM T51452 CJB1V2 11035207 EC50 = 247 nM T51452 C31EGD 11036467 EC50 = 268 nM T51452 CBV36I 11047145 EC50 = 202 nM T51452 C8B7TF 11067772 EC50 = 110 nM T51452 CAU9O6 11142977 EC50 = 84 nM T51452 CNSA17 11143256 EC50 = 245 nM T51452 CWO70Q 11673720 Ki = 24 nM T51452 CX7G9K 11759134 EC50 = 284 nM T51452 CL4XD0 11783674 EC50 = 20 nM T51452 CB9U0F 11825216 EC50 = 143 nM T51452 CTI32Y 15680235 EC50 < 100 nM T51452 CHBC95 23629662 Ki = 29.51 nM T51452 CN12BV 23629960 Ki = 7.413 nM T51452 CP4LU1 23630065 Ki = 2.239 nM T51452 CI50RV 25132065 Ki = 5.495 nM T51452 C47BLZ 25132069 Ki = 6.166 nM T51452 C8SR4O 25187292 IC50 = 271 nM T51452 CNC5G4 25187293 IC50 = 461 nM T51452 C6DBS4 25187295 IC50 = 57 nM T51452 CF1B8A 25188671 IC50 = 155 nM T51452 CW97NA 44273000 IC50 = 4 nM T51452 C5KV7A 44364531 EC50 = 879 nM T51452 CZK75V 44364548 EC50 = 459 nM T51452 C0FN6W 44364725 EC50 = 383 nM T51452 CYE1R8 44364726 EC50 = 55 nM T51452 CE8F3Y 44364734 EC50 = 327 nM T51452 COH5G6 44364735 EC50 = 134 nM T51452 C2VHW7 44364747 EC50 = 238 nM T51452 CZL2P0 44364907 EC50 = 70 nM T51452 CCX08E 44364918 EC50 = 256 nM T51452 C63IYQ 51003493 IC50 = 2114 nM T51452 CP8IG3 53317278 IC50 = 265 nM T51452 CP9I6O 53319883 IC50 = 472 nM T51452 CO6P3V 53320033 IC50 = 605 nM T51452 CCZ98L 53321188 IC50 = 213 nM T51452 C8MZR1 53322513 IC50 = 177 nM T51452 CTG2S9 53322514 IC50 > 3000 nM T51452 C29ARN 53323855 IC50 = 2 nM T51452 CBGD06 53323856 IC50 = 185 nM T51452 C9DJP1 53326435 IC50 = 154 nM T51452 C1JAV5 54581332 Ki = 10 nM T51452 C3XQ7U 54587225 Ki = 26.3 nM T51452 CJ8V6I 54587226 Ki = 56.23 nM T51452 C27YZH 88286432 Ki = 1000 nM T51452 CQ91VU 118278442 Ki = 32 nM T51452 CH0D4J 130439777 Ki = 360 nM T51452 C56XBU 130439778 Ki = 30000 nM T51452 C9N8LW 130439889 Ki = 789 nM T51452 D06SOQ 6918451 Ki = 0.58 nM T51452 D09IHE 6918583 Ki = 0.8 nM T51452 D0E7PY 11624499 Ki = 185 nM T51452 D0O9MG 5311203 Ki = 17 nM T78326 D0N1FS 26248 IC50 = 700 nM T78326 D0O1UZ 644019 IC50 > 100000 nM T78326 C3ERF2 30219 IC50 > 100000 nM T78326 C72VWJ 74288 IC50 = 19000 nM T78326 C7WN6M 80355 IC50 = 32000 nM T78326 CJ5T2N 98523 IC50 > 50000 nM T78326 CLOR58 154691 IC50 = 30 nM T78326 C2DF6O 160570 IC50 = 23000 nM T78326 CZ46HG 5315659 IC50 > 100000 nM T78326 C2AR0Z 6449999 IC50 > 50000 nM T78326 C29QMF 11055663 IC50 = 32000 nM T78326 C4CN3F 11601669 IC50 = 72300 nM T78326 CL58UG 20514378 IC50 = 10000 nM T78326 C80HKP 44398681 IC50 = 45000 nM T78326 C9KYX7 53689082 IC50 = 11000 nM T78326 CB70QO 57523549 IC50 = 7 nM T78326 C12DNA 59444416 IC50 > 100000 nM T78326 CYSZ16 70688797 IC50 = 314 nM T78326 CG8DY4 73291823 IC50 = 20 nM T78326 C57DRX 73291988 IC50 = 7 nM T78326 CDQC59 73294309 IC50 = 5 nM T78326 C5B8DQ 73356786 IC50 = 5 nM T78326 C53YHW 78319072 IC50 = 27 nM T78326 CB0RQ2 81689844 IC50 = 340 nM T78326 C12VNK 85872110 IC50 = 98000 nM T78326 C9-FEB-02 86274002 IC50 = 240 nM T78326 CI5F1D 86274233 IC50 = 100 nM T78326 C6K5EN 86274239 IC50 = 280 nM T78326 CR4ZJ2 86280724 IC50 = 1280 nM T78326 CR5G8K 86280727 IC50 = 71 nM T78326 CPC68B 86280729 IC50 = 8110 nM T78326 C74UGQ 86280860 IC50 = 9510 nM T78326 CWIM37 86280865 IC50 = 310 nM T78326 CD67QC 86280866 IC50 = 323 nM T78326 CKI68Y 86280867 IC50 = 140 nM T78326 CHZ7I6 86281014 IC50 = 2070 nM T78326 CV6ZO1 86281145 IC50 = 240 nM T78326 C26OXI 86281147 IC50 > 50000 nM T78326 CP1Q4G 86281282 IC50 = 17300 nM T78326 CPEG17 86281413 IC50 = 29360 nM T78326 CWN96H 86281416 IC50 = 25420 nM T78326 CRYE83 86281419 IC50 = 12910 nM T78326 C63SMU 86281538 IC50 = 1880 nM T78326 CROJ35 86281539 IC50 = 52 nM T78326 C3OEB4 86281540 IC50 = 76 nM T78326 C8RN9W 86281543 IC50 = 4470 nM T78326 CIQ5O3 86281544 IC50 = 160 nM T78326 CDYW71 86282210 IC50 = 122 nM T78326 CRO7N5 86282212 IC50 = 298 nM T78326 CIJ0U6 86282216 IC50 = 3110 nM T78326 C17RDC 86282353 IC50 = 1510 nM T78326 CH1XG7 86282354 IC50 = 2890 nM T78326 C93XIH 86282355 IC50 = 1110 nM T78326 C62EVZ 86282359 IC50 = 513 nM T78326 C05IOA 86282481 IC50 = 44 nM T78326 CV01AR 86282482 IC50 = 49 nM T78326 CNU9S3 86282483 IC50 = 33 nM T78326 CE2BL4 86282485 IC50 = 520 nM T78326 CXOJ45 86282487 IC50 = 37 nM T78326 CA7X5R 86282489 IC50 = 7 nM T78326 C7XS9W 86282624 IC50 = 12 nM T78326 CM3NV7 86282625 IC50 = 12830 nM T78326 CZ3DU9 86282626 IC50 = 30650 nM T78326 CEY75L 86282627 IC50 = 230 nM T78326 CM7C0T 86282766 IC50 = 73 nM T78326 CA5K3H 86700009 IC50 = 63 nM T78326 CGS6B3 86700028 IC50 = 302 nM T78326 CMO84Z 88924517 IC50 = 600 nM T78326 CVXD91 90424331 IC50 = 1040 nM T78326 C0ZNK5 90425119 IC50 = 250 nM T78326 CS91PZ 118727545 IC50 > 100000 nM T78326 CK9YC1 118727546 IC50 > 100000 nM T78326 CQ1MT5 118727547 IC50 > 100000 nM T78326 C6FP4M 118727548 IC50 > 100000 nM T78326 CSU24B 118727549 IC50 > 100000 nM T78326 CS15CM 118727550 IC50 > 100000 nM T78326 C1S6HU 118915486 IC50 = 2190 nM T78326 CL67PI 118915499 IC50 = 2670 nM T78326 CGU6N7 127025421 IC50 = 1720 nM T78326 CKI6R3 127029092 IC50 = 130 nM T78326 C9UFL8 132547272 IC50 = 20000 nM T78326 C6DA2U 132547273 IC50 = 38000 nM T78326 CH3MW2 132547274 IC50 = 78000 nM T78326 C38ZAQ 134130061 IC50 > 100000 nM T78326 CV5TF2 134145443 IC50 = 234 nM T78326 CR5V9U 134152906 IC50 = 507 nM T78326 CT8H0I 137632551 IC50 = 48 nM T78326 CU4EX8 137632575 IC50 = 1240 nM T78326 C6MSE9 137632802 IC50 = 10 nM T78326 CO36EY 137633578 IC50 = 167 nM T78326 CYM5W1 137633730 IC50 = 1983 nM T78326 CO1R2H 137634064 IC50 = 5070 nM T78326 C8VEN5 137635002 IC50 > 50000 nM T78326 C30ULI 137636190 IC50 = 31 nM T78326 COY74R 137637829 IC50 > 50000 nM T78326 CYEJ38 137640265 IC50 = 387 nM T78326 CXA46P 137640515 IC50 = 7180 nM T78326 CI76SB 137641029 IC50 = 39 nM T78326 CQY7R8 137641142 IC50 = 21 nM T78326 C9CM3B 137642349 IC50 = 2230 nM T78326 C86NAY 137645389 IC50 = 17 nM T78326 CAX26V 137645657 IC50 = 56 nM T78326 C6WJ4V 137645717 IC50 = 47690 nM T78326 CJI9O4 137647659 IC50 = 3010 nM T78326 C6H7UE 137647809 IC50 = 49 nM T78326 CBU65O 137653232 IC50 = 3470 nM T78326 C2CZK4 137653979 IC50 > 50000 nM T78326 CN2KJ7 137654116 IC50 = 15700 nM T78326 C3B1FX 137654484 IC50 = 88 nM T78326 C0DW7J 137655159 IC50 = 6 nM T78326 CSO9V7 137655498 IC50 = 17 nM T78326 C5SU2C 137657443 IC50 = 75 nM T78326 C6XEQ9 137658044 IC50 = 69 nM T78326 CGY1N8 137658817 IC50 = 187 nM T78326 CN2F8G 137658884 IC50 = 16 nM T78326 C3K2OT 137659365 IC50 = 6 nM T78326 CSUX67 137661910 IC50 = 23 nM T78326 CH37DX 137662244 IC50 = 133 nM T78326 C3T5LA 155522468 IC50 = 8000 nM T78326 D0D8PZ 93147 IC50 > 100000 nM T78326 D0U5LL 2543 IC50 > 50000 nM T78326 D0X3AT 44398718 IC50 = 17000 nM T74483 D0S6QR 214350 EC50 = 2400 nM T74483 D0W7IR 9887884 IC50 = 48 nM T74483 D0X7GL 121892 EC50 < 150 nM T74483 CNM41O 319496 IC50 = 1320 nM T74483 CYX02K 825799 IC50 > 30000 nM T74483 CX26LG 890442 EC50 = 743 nM T74483 CH83DC 2067822 EC50 = 800 nM T74483 C57RWN 2886850 IC50 = 14990 nM T74483 CRG0V9 4879449 IC50 = 12670 nM T74483 CY7EH6 7492195 EC50 = 1070 nM T74483 C03QJD 8232869 EC50 = 1750 nM T74483 C8QW3B 8232877 EC50 = 350 nM T74483 CBED14 9799604 EC50 = 1200 nM T74483 C14YJQ 18190094 EC50 = 2350 nM T74483 C4M9NP 24236861 EC50 = 950 nM T74483 CT3IK0 24247676 EC50 = 700 nM T74483 C9FZL6 24248347 IC50 = 163 nM T74483 CUV7D3 24684524 IC50 = 320 nM T74483 CI1G2C 26873419 IC50 = 70 nM T74483 C3S4BW 28015104 EC50 = 490 nM T74483 CN64WQ 44544347 IC50 = 1600 nM T74483 C2SOY1 46785920 IC50 > 30000 nM T74483 CFZ75O 46880148 IC50 > 30000 nM T74483 CL59YO 49852191 IC50 > 30000 nM T74483 C7ZUF5 49852192 IC50 > 30000 nM T74483 C6KX1V 49852195 IC50 > 30000 nM T74483 CD45TE 50898275 IC50 > 30000 nM T74483 CCOW18 50898276 IC50 = 5270 nM T74483 C8D5VY 50898278 EC50 > 30000 nM T74483 CZ86DL 51003787 IC50 > 30000 nM T74483 CO85BK 51003789 IC50 > 30000 nM T74483 CY25US 51003800 IC50 > 30000 nM T74483 C4WSV7 52914881 IC50 = 260 nM T74483 CR49FG 52914883 IC50 > 30000 nM T74483 C38YFR 52914885 IC50 = 210 nM T74483 CY8X7C 52914891 IC50 = 330 nM T74483 C32PZU 52914893 IC50 = 2220 nM T74483 C04IVY 52914895 EC50 = 990 nM T74483 CU7MH0 52914897 IC50 = 3500 nM T74483 C9MWG8 52914899 IC50 = 20230 nM T74483 CC1YE2 53313360 IC50 = 170 nM T74483 CJMR26 53313362 IC50 = 360 nM T74483 CEP5V0 53313364 IC50 = 330 nM T74483 CY93WA 53313366 IC50 = 130 nM T74483 C16IMX 53313368 IC50 = 470 nM T74483 C2UGL0 53313378 IC50 = 390 nM T74483 C58TGV 53313380 IC50 = 120 nM T74483 CN1X2Y 53313382 IC50 = 240 nM T74483 C78QHY 53313384 IC50 = 380 nM T74483 CY6T2X 53313386 IC50 = 280 nM T74483 CQM5U3 53313388 IC50 = 440 nM T74483 CNX2D9 53313390 EC50 = 170 nM T74483 CD42TV 53313393 EC50 = 1320 nM T74483 CBC81F 53313403 IC50 = 3310 nM T74483 CED9X4 53313407 EC50 = 1730 nM T74483 C6BL9E 53313474 IC50 > 30000 nM T74483 CQX6G3 53384811 EC50 = 1020 nM T74483 CZ0K3O 53384812 EC50 > 30000 nM T74483 CHJ85G 53384814 EC50 > 30000 nM T74483 C0MDO6 53384815 EC50 = 12270 nM T74483 CZ3BK9 53384824 EC50 = 27420 nM T74483 C8AH1W 53384828 EC50 = 7090 nM T74483 CB5O1N 53384829 EC50 > 30000 nM T74483 CD70RV 53384830 IC50 > 30000 nM T74483 CH7DP4 53384831 EC50 > 30000 nM T74483 CHI0N3 53384833 EC50 = 8660 nM T74483 CB2L5N 60200433 IC50 > 30000 nM T74483 C6LHX5 60200434 EC50 > 30000 nM T74483 CQC23I 73669559 EC50 = 1580 nM T74483 CK7DZ0 73670569 EC50 = 20 nM T74483 CN30SB 73670570 EC50 = 20 nM T74483 CXS6K4 73670740 EC50 = 34 nM T74483 CUR84N 73670742 EC50 = 330 nM T74483 C3QP0K 73671069 EC50 = 120 nM T74483 C24WCR 73671221 EC50 = 290 nM T74483 CGL1Q5 73671223 EC50 = 300 nM T74483 C0X7TP 73671695 EC50 = 130 nM T74483 C30OQS 73671696 EC50 = 220 nM T74483 CLZ1N0 123454460 EC50 = 250 nM T74483 CA2SK8 123554081 EC50 = 40 nM T74483 C4RBK5 123708382 EC50 = 1080 nM T74483 CHR7F1 123894154 EC50 = 2930 nM T74483 COB2A8 123898345 EC50 = 140 nM T74483 CX86QK 123944725 EC50 = 30 nM T74483 C30IVC 155491024 EC50 = 80 nM T74483 CTJ34I 155491025 EC50 = 630 nM T74483 C34WSD 155517409 IC50 = 5600 nM T74483 CLKU84 155519172 IC50 = 540 nM T74483 CCGZ20 155530937 IC50 = 160 nM T74483 CVBC47 155535120 IC50 = 200 nM T74483 CKA8V5 155536536 IC50 = 10000 nM T74483 D02BGR 9949648 EC50 = 690 nM T74483 D0FF6S 16038374 IC50 > 10000 nM T74483 D0P8PH 656732 IC50 = 55 nM T74483 D0W2FU 53347902 EC50 > 30000 nM T89515 D0T2IQ 443600 Ki = 0.3 nM T89515 C5MEC3 1736319 IC50 = 45000 nM T89515 C0LSJ1 9863482 IC50 = 8 nM T89515 C1F7RH 9864849 IC50 = 500 nM T89515 C2ZI6J 9904462 IC50 = 70 nM T89515 CZC32N 9905539 IC50 = 1 nM T89515 CO46AT 9978934 Ki = 19 nM T89515 C2YBW1 10384477 IC50 = 6 nM T89515 C23IFX 10445523 IC50 = 1040 nM T89515 CA74MQ 10456217 Ki = 2500 nM T89515 CKU12W 11244827 IC50 = 10 nM T89515 C3TP7Q 16057741 IC50 = 70 nM T89515 CN6E2R 16099871 IC50 = 200000 nM T89515 C36WFA 22096205 IC50 = 70 nM T89515 C2M0TF 44324304 IC50 = 20 nM T89515 CKNF72 44324347 IC50 = 50 nM T89515 CR51LS 44324348 IC50 = 40 nM T89515 C6LR3N 44324406 IC50 = 20 nM T89515 C5XRQ0 44324409 IC50 = 20 nM T89515 CVM73A 44324426 IC50 = 10 nM T89515 CX8M7N 44324427 IC50 = 50 nM T89515 C15HAD 44324519 IC50 = 20 nM T89515 C2CQ0K 44324520 IC50 = 30 nM T89515 CS97OG 44324562 IC50 = 20 nM T89515 CD2VX4 44324563 IC50 = 30 nM T89515 C4L6GE 44324567 IC50 = 1000 nM T89515 CM1US9 44324580 IC50 = 50 nM T89515 CZQJ43 44324610 IC50 > 1000 nM T89515 CCO0S7 44324611 IC50 = 200 nM T89515 CJB16T 44324659 IC50 = 30 nM T89515 CZQ0X8 44324677 IC50 = 600 nM T89515 C61KDH 44324687 IC50 = 100 nM T89515 CWMZ37 44339846 IC50 > 100000 nM T89515 C7ZA1O 44339862 IC50 > 100000 nM T89515 C39PEY 44339876 IC50 = 9910 nM T89515 CG2IT9 44339877 IC50 > 100000 nM T89515 C20TMG 44340129 IC50 = 8390 nM T89515 C8V9PJ 44345840 IC50 > 1000 nM T89515 CQ0FL7 44345845 IC50 > 1000 nM T89515 C3SD1F 44345873 IC50 = 200 nM T89515 CFV82Q 44345896 IC50 = 200 nM T89515 C1NC9U 44345897 IC50 > 1000 nM T89515 CS16FR 44345924 IC50 > 1000 nM T89515 CE9Y3L 44345990 IC50 > 1000 nM T89515 CE05IT 44345994 IC50 > 1000 nM T89515 C1WSP7 44418807 IC50 = 360000 nM T89515 CF2T6A 44418809 IC50 = 700000 nM T89515 CA3H4X 44418811 IC50 = 600000 nM T89515 CJTB64 44418813 IC50 = 250000 nM T89515 C4Z7YR 44418814 IC50 = 450000 nM T89515 C5TH6R 46944248 IC50 = 10000 nM T89515 CO47NY 49820157 IC50 = 59000 nM T89515 CPEM81 49820158 IC50 = 34000 nM T89515 CMRZ42 49820159 IC50 = 16000 nM T89515 C3W7RD 49820160 IC50 = 40000 nM T89515 C1V3ID 49820161 IC50 = 15000 nM T89515 C1URK4 49820162 IC50 = 15000 nM T89515 C1I6PE 49820310 IC50 = 65000 nM T89515 CW8O7L 49820311 IC50 = 6100 nM T89515 CKUJ18 49820312 IC50 = 25000 nM T89515 C1E7GJ 49820313 IC50 = 5200 nM T89515 CSCR58 49820936 IC50 = 32000 nM T89515 D0N8YA 159596 IC50 = 7 nM T63967 D0K0KH 656665 Ki = 55000 nM T63967 D0K7WK 4595 Ki = 46000 nM T63967 D0LM4A 170361 Ki = 0.06 nM T63967 D0Q9HF 187 EC50 = 1.7 nM T63967 D0T8GD 89594 Ki = 0.045 nM T63967 D0V8HA 4032 IC50 = 600 nM T63967 D0X4ZR 444 IC50 = 12000 nM T63967 D00EZO 10176607 Ki = 29 nM T63967 D01IVE 101616 Ki = 5.012 nM T63967 D05RSC 10131048 EC50 = 400 nM T63967 D08XPW 10235 Ki = 0.23 nM T63967 D0Y6OE 5310969 Ki = 0.04 nM T63967 D0ZC3C 5310985 Ki = 51 nM T63967 D0TF1E 9942427 EC50 = 5128.61 nM T63967 D00LVA 10176764 EC50 > 100000 nM T63967 D03UID 5310967 Ki = 25 nM T63967 D04HYP 3075702 Ki = 0.034 nM T63967 D09ADT 119380 EC50 = 10600 nM T63967 D0A5RD 9795056 IC50 = 20000 nM T63967 D0AB4Q 9824145 EC50 = 106 nM T63967 D0C9KD 44327552 Ki = 0.127 nM T63967 D0Q9RR 9794392 Ki = 140 nM T63967 D0Y9HH 3036156 EC50 = 320 nM T63967 C6GO7P 412 Ki = 29 nM T63967 CJ4M1W 1316 EC50 = 2500 nM T63967 C2IUD9 2181 Ki = 92 nM T63967 C45PUM 2551 Ki = 750 nM T63967 CP0J9N 3941 Ki = 90 nM T63967 C9IK1Y 4136 Ki = 23 nM T63967 C48GPY 5475 EC50 > 10000 nM T63967 C5H9CN 9287 Ki > 10000 nM T63967 CM3S5X 22124 EC50 = 41 nM T63967 C8G4LA 29758 Ki = 450 nM T63967 CL5WD4 67786 Ki = 30 nM T63967 C2NM4A 72503 IC50 = 62500 nM T63967 C0AMN5 84607 Ki = 20 nM T63967 CKI1H8 88393 Ki > 10000 nM T63967 CC3OR4 133106 EC50 = 2600 nM T63967 CL3I6A 165829 IC50 = 210 nM T63967 CVP7Y4 169017 Ki = 50 nM T63967 C2JM5W 202718 Ki = 160 nM T63967 CP81IV 204031 Ki > 31622.78 nM T63967 CT3Z4U 216066 EC50 = 10000 nM T63967 C89BMX 431734 Ki = 1.1 nM T63967 CI62ZN 442219 Ki = 600 nM T63967 C3IZC4 637026 IC50 = 150000 nM T63967 C4VX6K 637578 Ki > 31622.78 nM T63967 CK6SL0 666124 IC50 = 20600 nM T63967 C3LU7J 736282 Ki = 4 nM T63967 CN6V5X 852545 Ki > 10000 nM T63967 C03FIQ 902985 IC50 = 17100 nM T63967 CF42DT 1094969 IC50 = 21100 nM T63967 CR2T7N 1302023 IC50 = 13800 nM T63967 CS1DC9 1307388 IC50 = 7500 nM T63967 CA3E8R 1596080 Ki = 7000 nM T63967 CP2EN1 2064235 Ki = 6000 nM T63967 C6C7UX 2268445 IC50 = 19300 nM T63967 CIN1G2 2655600 IC50 = 4100 nM T63967 CHX06D 2995464 IC50 = 6000 nM T63967 CH81TW 3034748 Ki = 0.34 nM T63967 C3B1WI 3073763 Ki = 0.026 nM T63967 C3XM0R 3241687 IC50 = 9300 nM T63967 CAM0K9 3464560 IC50 = 13400 nM T63967 C9N6GB 3480598 IC50 = 23800 nM T63967 C9O7SE 3691150 IC50 = 8000 nM T63967 CHX01U 3945131 Ki > 10000 nM T63967 CHE9U8 4546524 IC50 = 7500 nM T63967 CSG73K 4694339 Ki = 0.04 nM T63967 CRC58X 4779153 IC50 = 10700 nM T63967 C1EVM7 5310971 IC50 > 2000000 nM T63967 C5FQ4L 5364095 Ki = 1600 nM T63967 CYB6T3 5835933 Ki = 1100 nM T63967 C95RIA 6412645 Ki = 4.1 nM T63967 CMK04Z 6433339 Ki > 3000 nM T63967 CF1NW5 6456944 IC50 = 14400 nM T63967 C69QWU 6471751 IC50 = 19600 nM T63967 C7M3WF 6472114 IC50 = 19400 nM T63967 CJ3FS9 6603935 IC50 = 500 nM T63967 CG5DH2 6604876 EC50 = 700 nM T63967 CLM7T3 6918622 IC50 = 5200 nM T63967 CUE4C9 7172378 Ki > 100000 nM T63967 CUN02J 7582345 IC50 = 6100 nM T63967 C81GRQ 8747436 IC50 = 14900 nM T63967 C50RLZ 8749430 IC50 = 17100 nM T63967 CZ69HA 9104895 IC50 = 9600 nM T63967 C08MRI 9794019 Ki = 1.1 nM T63967 C74CBS 9794141 EC50 = 750 nM T63967 C3R7GZ 9794155 EC50 = 1.622 nM T63967 CKI6W9 9794220 Ki = 2 nM T63967 CGC93J 9794354 EC50 = 1412.54 nM T63967 C0X9ZA 9794372 Ki = 0.15 nM T63967 C6EIV7 9794373 Ki = 0.13 nM T63967 CL15IQ 9807561 EC50 = 0.05 nM T63967 C2SHJ3 9812995 EC50 = 1400 nM T63967 C9YE1X 9813282 EC50 = 200 nM T63967 CF35HC 9813435 Ki = 1600 nM T63967 C6X3RP 9813490 Ki = 7 nM T63967 C9R8VP 9813576 EC50 = 900 nM T63967 C27UWZ 9813730 EC50 = 8709.64 nM T63967 CFLI74 9813803 EC50 = 269.15 nM T63967 CW0U8P 9815392 EC50 = 32359.37 nM T63967 CKTL63 9815484 EC50 = 1700 nM T63967 CBRU46 9815594 Ki = 0.27 nM T63967 C1M0SN 9815622 Ki = 1.4 nM T63967 C9GB1W 9815623 Ki > 500 nM T63967 C7FGY0 9815711 Ki = 100 nM T63967 CI7B0V 9815746 Ki = 0.75 nM T63967 CG4JD8 9815827 Ki = 4.9 nM T63967 CQS3E6 9815950 EC50 = 0.11 nM T63967 CN8HE1 9815968 EC50 = 3200 nM T63967 CS9G3F 9816020 Ki = 0.2 nM T63967 CXI84A 9816268 EC50 = 549.54 nM T63967 CLF78B 9816751 Ki = 0.1 nM T63967 CB8N5S 9817852 IC50 = 12000 nM T63967 C5OL1T 9834096 EC50 = 2691.53 nM T63967 CDF31X 9834107 Ki = 24 nM T63967 CHDY16 9834184 Ki = 2 nM T63967 C6FXS4 9834228 EC50 = 13489.63 nM T63967 C65DLA 9834234 EC50 = 9120.11 nM T63967 C80NVH 9834302 Ki = 0.44 nM T63967 C2D4HG 9834307 EC50 = 300 nM T63967 CO9DY5 9834308 EC50 = 537.03 nM T63967 CQY34E 9834353 EC50 = 1930 nM T63967 CQ98AW 9834452 EC50 = 23.99 nM T63967 CG6D1L 9834532 Ki = 0.12 nM T63967 C1VRA6 9834541 Ki = 34 nM T63967 C0JWH4 9834547 Ki = 264 nM T63967 CUB3G9 9834620 EC50 = 134 nM T63967 C4I1SM 9834864 EC50 = 4073.8 nM T63967 C7YM1O 9834889 Ki = 0.3 nM T63967 C82IBV 9835659 IC50 = 1.413 nM T63967 C6QUC8 9835715 Ki = 3.1 nM T63967 C7BZE2 9836977 EC50 = 720 nM T63967 C68OVP 9836984 Ki = 90 nM T63967 CJW79D 9836998 EC50 = 30902.95 nM T63967 CB4UO0 9837143 EC50 = 850 nM T63967 CJ2X8T 9837259 Ki = 200 nM T63967 C7V1AH 9837340 EC50 = 25000 nM T63967 C5R9OC 9837377 EC50 = 11000 nM T63967 COT0X4 9837478 Ki = 0.31 nM T63967 C9GDO4 9837582 Ki = 0.15 nM T63967 C95UWI 9837971 EC50 = 370 nM T63967 CU9I1H 9838143 Ki = 39 nM T63967 CJ7CI4 9855608 EC50 = 1819.7 nM T63967 C4MG8D 9855694 EC50 = 407.38 nM T63967 CBSF19 9855936 EC50 = 1096.48 nM T63967 CZS71O 9855966 EC50 = 600 nM T63967 C10LFH 9856458 EC50 = 176 nM T63967 CZB45J 9856887 EC50 = 323.59 nM T63967 CF50CE 9856916 Ki = 370 nM T63967 CTND15 9859046 Ki = 0.16 nM T63967 C1EU9Q 9859868 Ki = 13 nM T63967 CV3R4A 9860762 Ki < 5 nM T63967 CYL5G3 9877467 Ki > 10000 nM T63967 CB6Z8S 9877653 EC50 = 4897.79 nM T63967 CSP4D2 9877707 EC50 = 3388.44 nM T63967 CFO4D6 9877782 EC50 = 2187.76 nM T63967 CT9M8Z 9877804 Ki = 75 nM T63967 CK03PX 9877833 Ki = 13 nM T63967 CX56YU 9878090 IC50 = 181.97 nM T63967 C9EKX4 9878102 Ki = 1.9 nM T63967 CFZ76C 9878279 Ki = 0.19 nM T63967 CQ8AG6 9878601 EC50 = 16982.44 nM T63967 C34MOW 9881232 EC50 = 4265.8 nM T63967 CK9M6R 9881718 Ki = 0.33 nM T63967 CLWT60 9882021 EC50 = 3200 nM T63967 C5XW1U 9883385 EC50 = 0.036 nM T63967 C7LD1U 9899354 EC50 = 37.15 nM T63967 CRST76 9899814 Ki = 0.2 nM T63967 CF51PO 9900094 Ki = 0.28 nM T63967 CV3BX9 9900445 Ki = 0.75 nM T63967 C8E0IP 9900637 IC50 = 1.413 nM T63967 CS81KW 9904090 Ki = 34 nM T63967 CX73LN 9917490 IC50 = 9200 nM T63967 CAJ1X8 9920686 Ki = 0.1 nM T63967 CFJR18 9920831 Ki = 13 nM T63967 CB8CG3 9920836 Ki = 14 nM T63967 CDJ34P 9921125 Ki = 0.36 nM T63967 CTE89G 9921869 EC50 = 851.14 nM T63967 CIQ1Z2 9925774 Ki = 0.018 nM T63967 C07SPN 9942280 Ki = 1700 nM T63967 CAV98S 9942481 EC50 = 22908.68 nM T63967 CVYM29 9942613 EC50 = 7690 nM T63967 C8ETL1 9942787 EC50 = 75.86 nM T63967 CO2N0J 9943498 IC50 = 229.09 nM T63967 C6AZ3X 9943908 IC50 = 3300 nM T63967 CNB64Y 9944799 Ki = 200 nM T63967 CY2Q8J 9964230 EC50 = 1600 nM T63967 CZE08N 9964805 EC50 = 263.03 nM T63967 CBP36J 9964897 Ki > 500 nM T63967 CR80UF 9965385 Ki = 0.14 nM T63967 CFZ9D7 9972515 IC50 = 9800 nM T63967 COP08X 9972881 IC50 = 11000 nM T63967 C4Q5YW 9996559 Ki > 10000 nM T63967 CIWG38 10015966 Ki = 2600 nM T63967 CID3J4 10019186 Ki > 10000 nM T63967 C4BE2Y 10025698 Ki = 0.09 nM T63967 C8BM4D 10044336 Ki = 300 nM T63967 C6XFH7 10058322 EC50 = 70.79 nM T63967 CGM3W9 10059716 Ki = 10 nM T63967 C7O5DA 10061682 Ki = 14000 nM T63967 CJ6B2U 10081505 EC50 = 416.87 nM T63967 CL9EM5 10081731 EC50 = 2100 nM T63967 COE53P 10082341 EC50 = 12.88 nM T63967 CE64SB 10083372 IC50 = 640 nM T63967 CUW85L 10085732 EC50 > 100000 nM T63967 CX4AG8 10087431 Ki > 10000 nM T63967 CZBI21 10107007 Ki = 0.47 nM T63967 CCZ3T9 10130346 Ki = 0.28 nM T63967 CN0BQ7 10130391 EC50 = 977.24 nM T63967 CTV58J 10130408 Ki = 0.17 nM T63967 C2CT5D 10130418 Ki = 32 nM T63967 CDH4J3 10130527 Ki = 2.2 nM T63967 C6LB2N 10130752 Ki = 0.39 nM T63967 C7TQN9 10131290 EC50 = 64.57 nM T63967 CN4L0G 10154205 IC50 = 100 nM T63967 C15FVX 10154254 Ki = 1.6 nM T63967 C63VHC 10154344 Ki = 0.5 nM T63967 CY64SL 10176226 Ki = 5.8 nM T63967 CN05GL 10176454 Ki = 1 nM T63967 CM9B2Z 10176482 Ki = 6.5 nM T63967 CR2DG8 10176616 EC50 = 19952.62 nM T63967 C0I2BK 10176727 Ki = 0.1 nM T63967 C1X0LJ 10176791 Ki = 6.5 nM T63967 CL4R8D 10198017 EC50 = 2600 nM T63967 C1F2DC 10198406 EC50 = 180 nM T63967 C7J4YE 10198642 Ki = 0.55 nM T63967 C6TFO1 10219646 Ki = 2.8 nM T63967 CM58IK 10219887 EC50 = 3000 nM T63967 CLMB50 10219900 EC50 = 5700 nM T63967 CBS1I4 10219939 Ki = 0.182 nM T63967 C8QE2I 10220229 EC50 = 4365.16 nM T63967 CL5ZJ2 10243433 EC50 = 91.2 nM T63967 C7L5PB 10246574 Ki = 1300 nM T63967 CN2JQ8 10262309 EC50 > 100000 nM T63967 C7X5QD 10263121 EC50 = 1400 nM T63967 CX8B5S 10267729 EC50 > 10000 nM T63967 CZP3L6 10313455 Ki = 2.9 nM T63967 CV3L6Y 10321902 Ki = 0.14 nM T63967 CJT2H9 10359708 Ki > 10000 nM T63967 C5AN1L 10375812 EC50 = 162.18 nM T63967 CDE3N9 10402507 IC50 = 0.871 nM T63967 CLC49H 10421899 Ki = 32 nM T63967 CNY59C 10443079 EC50 = 24.55 nM T63967 CHR72Q 10443815 Ki = 29 nM T63967 C8BCV0 10465833 EC50 = 1900 nM T63967 C1B7AQ 10488548 IC50 = 1.905 nM T63967 C8TPU0 10510985 Ki = 2285 nM T63967 CKE8Q0 10559695 EC50 = 141.25 nM T63967 C4GLK8 10559857 EC50 = 22908.68 nM T63967 CPQ7O4 10560219 EC50 = 4800 nM T63967 C2M0FI 10582927 Ki = 47 nM T63967 CM2U3Q 10607315 Ki = 34 nM T63967 CY7I8H 10608955 EC50 = 12882.5 nM T63967 C32BYZ 10639739 Ki = 2.2 nM T63967 C8X0BP 10654371 Ki ~ 6000 nM T63967 CYCQ03 10654891 EC50 = 229.09 nM T63967 CRFH56 10656505 EC50 = 1096.48 nM T63967 C7BYI3 10679307 Ki = 212 nM T63967 CPF17I 10704502 EC50 = 3630.78 nM T63967 C7OJ0S 10726068 Ki = 22 nM T63967 CPU24S 10727034 EC50 = 10964.78 nM T63967 CYDA95 10753258 IC50 = 2.399 nM T63967 CU4QZ7 10799900 IC50 = 169.82 nM T63967 C2RSE8 10880951 Ki = 16900 nM T63967 C0FN1U 10922391 Ki = 8.3 nM T63967 CJM0E5 10924232 EC50 = 39810.72 nM T63967 CZR3T6 10932563 IC50 = 600 nM T63967 CC97MS 10956816 Ki = 110 nM T63967 CIDQ52 10957379 Ki = 300 nM T63967 CC7PU4 11064290 Ki = 820 nM T63967 CWB47N 11086486 Ki = 95800 nM T63967 CLD5Z0 11098414 IC50 = 3400 nM T63967 C8O5VS 11119032 Ki = 110 nM T63967 C0X9JF 11162968 Ki > 20000 nM T63967 CO83JA 11183894 IC50 = 5100 nM T63967 CPVA01 11255359 IC50 = 15000 nM T63967 CXH8G3 11278436 IC50 = 11000 nM T63967 CPU14O 11288721 EC50 = 5950 nM T63967 CC9Q3V 11332920 Ki = 94 nM T63967 CU1S6Y 11400044 IC50 = 27.8 nM T63967 C57YWO 11422871 IC50 = 20.8 nM T63967 C08TAW 11458897 Ki > 31622.78 nM T63967 CP1WH5 11461365 EC50 > 100000 nM T63967 CF5R1Z 11463970 IC50 = 15000 nM T63967 C9L2AH 11474847 IC50 = 942000 nM T63967 CP8QT3 11493499 EC50 = 7585.78 nM T63967 CVZ02O 11499356 EC50 = 36.31 nM T63967 CP52OD 11514075 IC50 = 1 nM T63967 CCE92P 11515142 IC50 = 0.3802 nM T63967 C9AWJ0 11516571 EC50 = 1.288 nM T63967 C1A8LW 11523132 EC50 = 2089.3 nM T63967 CT1XJ7 11528487 EC50 = 25000 nM T63967 C6E9WD 11543033 EC50 = 26915.35 nM T63967 CU54BI 11550362 EC50 = 169.82 nM T63967 CO29QA 11573965 IC50 = 21.88 nM T63967 COJH10 11596787 IC50 = 0.6457 nM T63967 C6GU8D 11615990 EC50 = 181.97 nM T63967 CN4Z5C 11679149 IC50 = 25118.86 nM T63967 CIQ12L 11701287 Ki = 0.36 nM T63967 CA1C9Y 11715647 EC50 > 100000 nM T63967 C02EFG 11832145 Ki = 5400 nM T63967 CB34AR 11957729 Ki = 7800 nM T63967 CT76NQ 12086849 EC50 = 13 nM T63967 CF96QD 12303261 IC50 = 1570 nM T63967 CLJ14R 12358972 IC50 = 500 nM T63967 C0IJV5 12392828 IC50 = 6900 nM T63967 CE5X1A 12625600 Ki = 7.9 nM T63967 C5UK2P 13996231 EC50 = 5500 nM T63967 C17ZBV 14262870 Ki = 910 nM T63967 C6EO2H 14262872 Ki = 10000 nM T63967 CHL5U6 14279649 Ki = 170 nM T63967 CKJN91 14279657 Ki = 120 nM T63967 CE5FB3 14626249 Ki = 470 nM T63967 C3IV5B 14806309 IC50 = 36.6 nM T63967 C4L0PS 15114748 Ki = 5700 nM T63967 C4YD8Q 15521852 Ki = 3330 nM T63967 CB4OC5 15521853 Ki = 1260 nM T63967 CVP7D8 15753505 Ki = 60 nM T63967 C7LF3K 16099069 EC50 = 330 nM T63967 CJLU49 16099070 EC50 = 1000 nM T63967 CJH4F0 16099071 EC50 = 12 nM T63967 C52LBH 16099072 EC50 = 7.762 nM T63967 CXN75R 16099073 EC50 = 7.2 nM T63967 CGU63X 16099074 EC50 = 128.82 nM T63967 C4FEW3 16099075 EC50 = 2187.76 nM T63967 C6OR8V 16099076 EC50 = 4980 nM T63967 C91AUD 16099077 EC50 = 1348.96 nM T63967 C21YIA 16099078 EC50 = 100 nM T63967 CXD7Z3 16099079 EC50 = 20.89 nM T63967 C0WZR4 16099080 EC50 = 6.1 nM T63967 CLR21F 16099081 EC50 = 1690 nM T63967 CQ0C2P 16099082 EC50 = 172 nM T63967 CUI8P1 16099083 EC50 = 338.84 nM T63967 C9PRA2 16099084 EC50 = 350 nM T63967 CI5K4R 16099085 EC50 = 78.3 nM T63967 C0GV4U 16099091 EC50 = 75.86 nM T63967 C83HRV 16099099 EC50 = 150 nM T63967 CFV86M 16099100 EC50 = 81.28 nM T63967 CVN2J3 16099101 EC50 = 46.77 nM T63967 CC9DA0 16099102 EC50 = 1900 nM T63967 CQS1C4 16099103 EC50 = 2691.53 nM T63967 CDQF19 16099104 EC50 = 616.6 nM T63967 C3K8CO 16099105 EC50 = 645.65 nM T63967 CWB4P7 16099106 EC50 = 109.65 nM T63967 CJ1P6E 16099107 EC50 = 360 nM T63967 CM9G0S 16099108 EC50 = 180 nM T63967 CU5J2I 16099109 EC50 = 213.8 nM T63967 C7S1GW 16099110 EC50 = 199.53 nM T63967 CZB59V 16099111 EC50 = 109 nM T63967 CZ94VM 16099112 EC50 = 1479.11 nM T63967 C2EIJ5 16099113 EC50 = 8420 nM T63967 CL5CR3 16099114 EC50 = 4390 nM T63967 C9XZI4 16099115 EC50 = 359 nM T63967 CO8ID2 16126643 IC50 = 5360 nM T63967 CGZN70 16637618 Ki = 17 nM T63967 C9O4RE 16727410 Ki = 1200 nM T63967 CI49EV 16747994 Ki = 0.15 nM T63967 CLC3F4 16748111 Ki = 0.02 nM T63967 CHT0S5 17384430 IC50 = 13900 nM T63967 C1OTB6 18177037 Ki = 920 nM T63967 C3XHW0 18180401 EC50 > 10000 nM T63967 C5H8PA 18432673 EC50 = 70.79 nM T63967 C1HOU8 18432695 EC50 = 1584.89 nM T63967 CFWM01 20396098 Ki = 1.1 nM T63967 C47LEX 20430515 Ki = 360 nM T63967 CF81LI 20669017 Ki = 65.2 nM T63967 CXQM78 20695745 IC50 > 100 nM T63967 CCO62K 21124461 Ki > 31622.78 nM T63967 COM7F5 21309700 EC50 > 1000000 nM T63967 C4PJN6 21574409 Ki = 0.763 nM T63967 CABE87 21833117 Ki = 3390 nM T63967 C0EO2W 22215312 Ki = 34 nM T63967 C6EX4B 22291236 EC50 > 100000 nM T63967 C5ZCN8 22872635 Ki = 0.14 nM T63967 CSJD40 22987731 EC50 = 4 nM T63967 COJ4U7 22987762 EC50 = 1.1 nM T63967 CP7MK3 22987764 EC50 > 100 nM T63967 CR5B8K 22987817 EC50 > 100 nM T63967 CXWI74 23332842 EC50 > 100000 nM T63967 CW2R4M 23624283 IC50 = 5011.87 nM T63967 CBQS32 23634540 EC50 = 912.01 nM T63967 CI4GY6 23634543 EC50 = 200 nM T63967 CZC61E 23634545 EC50 = 724.44 nM T63967 C2P6RE 23634548 EC50 = 43.65 nM T63967 C59MUH 23634670 EC50 = 72.44 nM T63967 CJY49C 23634788 EC50 = 30902.95 nM T63967 CBS3A5 23634911 EC50 = 676.08 nM T63967 CSYC96 23634914 EC50 = 1100 nM T63967 C4CR5U 23634916 EC50 = 1174.9 nM T63967 CQUI19 23635035 EC50 = 389.05 nM T63967 C2GAQ9 23635037 EC50 = 2187.76 nM T63967 CH2O4E 23635039 EC50 = 6760.83 nM T63967 CUB17S 23635157 EC50 = 300 nM T63967 CM19ZP 23635159 EC50 = 10000 nM T63967 C1H7CZ 23635160 EC50 = 1548.82 nM T63967 CIK9U8 23635162 EC50 = 1174.9 nM T63967 C5KOC7 23635288 EC50 = 776.25 nM T63967 CYFB26 23635289 EC50 = 4570.88 nM T63967 C15KIQ 23635417 EC50 = 7244.36 nM T63967 CVD51I 23635423 EC50 = 1479.11 nM T63967 CD94YA 23635530 EC50 = 3801.89 nM T63967 CCJ24W 23635651 EC50 = 295.12 nM T63967 CRE52L 23635654 EC50 = 6165.95 nM T63967 CI8VQ9 23635786 EC50 = 13182.57 nM T63967 CX52UA 23636037 EC50 = 41.69 nM T63967 CG2D4Y 23636156 EC50 = 2041.74 nM T63967 C2X7UR 23636160 EC50 = 500 nM T63967 CB18JU 23636165 EC50 = 147.91 nM T63967 CMI29X 23636510 EC50 = 1071.52 nM T63967 CDKB19 23636512 EC50 = 9332.54 nM T63967 C2JG3M 23636514 EC50 = 13182.57 nM T63967 CW02CY 23643977 IC50 > 10000 nM T63967 C3QEI4 24686533 IC50 = 13600 nM T63967 CE2XP4 24795080 Ki = 30 nM T63967 CZD45C 24894145 EC50 = 18 nM T63967 C84AQE 24945028 Ki = 33 nM T63967 CHY7C1 24945029 Ki = 32 nM T63967 CV07CE 24945030 Ki = 42 nM T63967 C30XMU 24945031 Ki = 2 nM T63967 CGI46H 24945032 Ki = 2 nM T63967 C50QZG 24945033 Ki = 74 nM T63967 CT13LF 24945123 Ki = 19 nM T63967 CI0YH2 24945124 Ki = 340 nM T63967 C3WIQ9 24945126 Ki = 110 nM T63967 C93SUY 24945129 Ki = 49 nM T63967 C5MNT9 24945296 Ki = 67 nM T63967 C78HXO 24945297 Ki = 20 nM T63967 CY5D6P 24945298 Ki = 190 nM T63967 C1T0FO 24945299 Ki = 46 nM T63967 C3UP8T 24945300 Ki = 15 nM T63967 CKJG57 24945301 Ki = 5 nM T63967 CW9F1R 24945302 Ki = 23 nM T63967 C0N7YV 24945376 Ki = 26 nM T63967 C3LBH5 24945542 Ki = 37 nM T63967 CRYT93 24970319 Ki = 8 nM T63967 CWM0S4 24998996 Ki > 10000 nM T63967 CKN91Y 24999304 Ki > 10000 nM T63967 C3D4RY 25001268 Ki > 10000 nM T63967 C84OCG 25001269 Ki > 10000 nM T63967 C21TAX 25009380 Ki > 10000 nM T63967 CJD7A3 25009564 Ki > 10000 nM T63967 CZN8O6 25009747 Ki > 10000 nM T63967 CKSD03 25009944 Ki > 10000 nM T63967 CD2CK3 25085910 IC50 = 145000 nM T63967 CQR84M 25147644 Ki = 1700 nM T63967 CI1V6B 25155668 Ki = 96 nM T63967 C9U2QX 25156769 Ki = 28000 nM T63967 CCB91S 25182691 Ki = 1300 nM T63967 CF4OQ9 25182692 Ki = 1300 nM T63967 C06EBO 27185027 IC50 = 12400 nM T63967 CY1I9X 29354120 IC50 = 8000 nM T63967 CGKR74 37066353 IC50 = 20300 nM T63967 C0DJ8H 39010244 IC50 > 100000 nM T63967 C1CWU0 42631007 IC50 = 7943.28 nM T63967 CFU84B 42636894 IC50 = 460 nM T63967 CJV6A7 44158944 IC50 = 3800 nM T63967 C7BU8N 44190125 EC50 = 40 nM T63967 CR80FS 44190223 EC50 = 370 nM T63967 CB4K5O 44190326 EC50 > 100000 nM T63967 C83NGA 44190552 EC50 > 100000 nM T63967 C6NT5U 44190553 EC50 > 100000 nM T63967 C6TOC5 44199430 Ki = 12 nM T63967 C43GIX 44222896 Ki = 8 nM T63967 CBP9G1 44222951 Ki = 1 nM T63967 CN9CA4 44223026 Ki = 38 nM T63967 C6MCF2 44223074 Ki = 4 nM T63967 CG5Q6P 44223132 Ki = 20 nM T63967 CNP36F 44224169 EC50 = 2500 nM T63967 CCW0G6 44225415 Ki = 157 nM T63967 CK7F2E 44240743 IC50 > 30000 nM T63967 C4W0SH 44247585 EC50 > 100000 nM T63967 C7V0WO 44297526 Ki = 0.05 nM T63967 CD74SQ 44297578 Ki > 1000 nM T63967 C1RJ4O 44297660 Ki = 0.3 nM T63967 CGUR82 44297661 Ki = 3.2 nM T63967 CJ7I3W 44297672 Ki > 1000 nM T63967 CJ2M9Q 44299190 Ki = 0.027 nM T63967 CKM8H4 44304543 EC50 = 1000 nM T63967 CP83TA 44304625 EC50 = 42 nM T63967 CLA5P6 44304691 EC50 = 2.2 nM T63967 CT6PM2 44311174 EC50 = 1202.26 nM T63967 CH7MV5 44318740 IC50 = 3200 nM T63967 CIR5C3 44318904 EC50 = 2200 nM T63967 CK6X5A 44318972 EC50 > 1000000 nM T63967 CUZ6R3 44318995 EC50 = 1000 nM T63967 C01YXZ 44319012 EC50 = 2300 nM T63967 CD10NQ 44319160 EC50 = 2600 nM T63967 CTMR48 44324442 Ki = 7.4 nM T63967 CZ28JL 44324548 EC50 > 1000000 nM T63967 CF2YA4 44324564 EC50 = 11000 nM T63967 CZ1K7J 44328413 Ki = 170 nM T63967 C7URA4 44328470 Ki = 2.6 nM T63967 C0L7IN 44328663 Ki = 40 nM T63967 CSQ6B7 44328681 Ki = 120 nM T63967 CUQC95 44340717 Ki = 450 nM T63967 CC7D2K 44346647 Ki = 330 nM T63967 CHYG84 44346866 Ki > 10000 nM T63967 CZ2E0P 44346902 Ki > 10000 nM T63967 CQ32XS 44346903 Ki > 10000 nM T63967 CT42RA 44346914 Ki > 10000 nM T63967 C5R4WQ 44348072 IC50 = 5495.41 nM T63967 CE6U1G 44348090 IC50 = 8000 nM T63967 C8RAO6 44348296 IC50 = 13500 nM T63967 COA40Y 44348309 IC50 = 5011.87 nM T63967 CR42HE 44348319 IC50 = 6309.57 nM T63967 C4XKW0 44348376 IC50 = 4897.79 nM T63967 C0SOG1 44348388 IC50 = 7943.28 nM T63967 CVGZ81 44348389 IC50 = 9332.54 nM T63967 CRC25U 44354684 EC50 = 1870 nM T63967 CGY76Q 44365978 Ki > 10000 nM T63967 CG5I6B 44365979 Ki = 470 nM T63967 CE2WX5 44366124 Ki = 154 nM T63967 C5KL2H 44366125 Ki > 10000 nM T63967 CH3VS0 44395275 Ki = 0.771 nM T63967 C1H7FD 44398087 IC50 = 9.6 nM T63967 CNL4B1 44398091 IC50 = 0.75 nM T63967 C1C3EN 44398092 IC50 = 1.5 nM T63967 CYOE97 44399319 Ki = 5.7 nM T63967 C6TRQ8 44399348 Ki > 500 nM T63967 CZ42OX 44399413 Ki = 72 nM T63967 CZFD84 44399504 Ki > 500 nM T63967 C0ZWQ4 44399533 Ki > 500 nM T63967 C6HKB4 44399550 Ki > 500 nM T63967 CK8AS7 44401289 Ki > 10000 nM T63967 CS0GU1 44401325 Ki > 10000 nM T63967 CU1C5A 44401533 Ki > 10000 nM T63967 C4NL5E 44401629 Ki > 10000 nM T63967 CL76NW 44401675 Ki > 10000 nM T63967 C4Z6KV 44401680 Ki > 10000 nM T63967 CGTU10 44401691 Ki > 10000 nM T63967 C6TJ5V 44401698 Ki > 10000 nM T63967 C9O8UH 44401699 Ki > 10000 nM T63967 C9CWB7 44401706 Ki > 10000 nM T63967 CP65LR 44401721 Ki > 10000 nM T63967 C6WF5T 44401722 Ki > 10000 nM T63967 CPXL47 44401738 Ki > 10000 nM T63967 C1KT6I 44401740 Ki > 10000 nM T63967 C8Q6ET 44401749 Ki > 10000 nM T63967 CD7HT3 44401750 Ki > 10000 nM T63967 CR7IO2 44401761 Ki > 10000 nM T63967 C2DE3R 44401766 Ki > 10000 nM T63967 C5ZE8B 44401777 Ki > 10000 nM T63967 CMI78Q 44401778 Ki > 10000 nM T63967 C7VS2K 44401780 Ki > 10000 nM T63967 CHDC82 44401785 Ki > 10000 nM T63967 CC18BW 44401791 Ki > 10000 nM T63967 C9ATN1 44401792 Ki > 10000 nM T63967 C5K4IQ 44401800 Ki > 10000 nM T63967 C25OJD 44401806 Ki > 10000 nM T63967 C01RPV 44401821 Ki > 10000 nM T63967 C8MVZ7 44401829 Ki > 10000 nM T63967 C8ZU9E 44401866 Ki > 10000 nM T63967 C56MID 44401877 Ki > 10000 nM T63967 CUEJ14 44401878 Ki > 10000 nM T63967 CETN06 44401885 Ki > 10000 nM T63967 CYWJ71 44401891 Ki > 10000 nM T63967 C6MHU9 44401893 Ki > 10000 nM T63967 CR3X4T 44401897 Ki > 10000 nM T63967 C10FNX 44401906 Ki > 10000 nM T63967 CSRJ78 44401907 Ki > 10000 nM T63967 COH39X 44401927 Ki > 10000 nM T63967 C0B6GX 44401939 Ki > 10000 nM T63967 C1D7FJ 44401940 Ki > 10000 nM T63967 CR3TJ9 44401942 Ki > 10000 nM T63967 CG7SY1 44401944 Ki > 10000 nM T63967 CRAB67 44401955 Ki > 10000 nM T63967 C0V9BW 44401970 Ki > 10000 nM T63967 C9FB0N 44401980 Ki > 10000 nM T63967 CV67RU 44401983 Ki > 10000 nM T63967 CC25UQ 44401984 Ki > 10000 nM T63967 CN3P4D 44401986 Ki > 10000 nM T63967 CXN8Q9 44402005 Ki > 10000 nM T63967 CN9C1P 44402006 Ki > 10000 nM T63967 CPIO37 44402059 Ki > 10000 nM T63967 CL7TW8 44402150 Ki > 10000 nM T63967 C7GV8I 44402194 Ki > 10000 nM T63967 C6CAO3 44402258 Ki > 10000 nM T63967 CQL3U1 44402277 Ki > 10000 nM T63967 CZTQ12 44404455 Ki = 2 nM T63967 CN37JP 44419364 Ki = 0.0785 nM T63967 C20KPD 44423688 Ki = 2500 nM T63967 CLQ56U 44427060 EC50 = 275.42 nM T63967 C9QSB5 44427064 EC50 = 7413.1 nM T63967 CF4O6R 44427071 EC50 = 1500 nM T63967 C8DAS2 44436056 Ki = 128 nM T63967 CY7UK0 44436057 Ki = 12400 nM T63967 CDQG71 44436059 Ki = 7370 nM T63967 CW6K3G 44436062 Ki = 17.2 nM T63967 C1JNK4 44442621 IC50 = 3500 nM T63967 C7WOJ8 44442623 IC50 = 2500 nM T63967 C12XGE 44456400 Ki > 10000 nM T63967 C5Q3NI 44542504 IC50 = 35 nM T63967 CYX7H5 44542510 IC50 = 9.2 nM T63967 C71QGD 44542511 IC50 = 19 nM T63967 C2EDU6 44542955 IC50 = 32 nM T63967 C03MXJ 44543264 IC50 = 45 nM T63967 CL5UK7 44543265 IC50 = 32 nM T63967 C6S4JY 44565060 Ki = 7.6 nM T63967 CM8U6J 44570006 Ki = 12000 nM T63967 CH84MQ 44570007 Ki = 23000 nM T63967 C2E3LJ 44570008 Ki = 125.89 nM T63967 CWPR65 44570009 Ki = 1900 nM T63967 C13RLY 44570010 Ki = 36 nM T63967 CIV69B 44570011 Ki = 48 nM T63967 CG4YE9 44570012 Ki = 199.53 nM T63967 C0ZL8N 44570053 Ki = 1100 nM T63967 CQ4K3T 44570054 Ki = 6309.57 nM T63967 CVGP31 44570055 Ki = 290 nM T63967 CPST94 44570056 Ki = 1500 nM T63967 C0VZ9I 44570057 Ki = 91 nM T63967 CQ8L9B 44570097 Ki = 1584.89 nM T63967 CU7S2P 44570098 Ki = 100000 nM T63967 CFUE82 44570099 Ki = 300000 nM T63967 C31CSH 44570100 Ki = 3600 nM T63967 CQS02B 44570101 Ki = 6309.57 nM T63967 CMP1K2 44570102 Ki = 39810.72 nM T63967 C2X4GC 44570103 Ki = 31622.78 nM T63967 C18JSV 44570104 Ki = 1584.89 nM T63967 C7I6OB 44570105 Ki = 9800 nM T63967 C1A2TU 44575473 Ki > 10000 nM T63967 CECB52 44577577 Ki = 0.46 nM T63967 C97DTY 44580092 EC50 = 230 nM T63967 C4VZA0 44580093 EC50 = 200 nM T63967 CXH64K 44580094 EC50 = 130 nM T63967 CI29TB 44580095 EC50 = 410 nM T63967 CWU9E3 44580096 EC50 = 1300 nM T63967 CQG3J7 44580171 EC50 = 4600 nM T63967 CU97PQ 44580172 EC50 = 33 nM T63967 CYZ19X 44580173 EC50 = 12 nM T63967 CRX95K 44580174 EC50 = 3 nM T63967 CC0B3Q 44580175 EC50 = 34 nM T63967 C5LVN7 44580251 EC50 = 350 nM T63967 C5Y3MD 44580252 EC50 = 120 nM T63967 CP63YN 44580284 EC50 = 100000 nM T63967 C9YRF5 44580285 EC50 = 1200 nM T63967 CBO1H3 44580286 EC50 = 48 nM T63967 CEL61G 44580287 EC50 = 6 nM T63967 CQN2R7 44580288 EC50 = 270 nM T63967 CB7K9C 44580289 EC50 = 220 nM T63967 C6E9SG 44580290 EC50 = 3 nM T63967 CVH9T3 44593550 Ki = 13 nM T63967 C5N9PS 44719858 EC50 = 10000 nM T63967 CJY9C4 45115751 Ki = 0.4 nM T63967 C7MB5N 45141377 IC50 = 37 nM T63967 CMSH89 45141378 IC50 = 36 nM T63967 CTL0U6 45141609 IC50 > 100 nM T63967 CRU4W0 45254040 EC50 = 10.2 nM T63967 CQK28Z 45379093 Ki = 12 nM T63967 CK6X3B 45786849 Ki = 1.6 nM T63967 CVCY62 46191141 EC50 = 1560 nM T63967 C6G2TZ 46191426 IC50 = 31.62 nM T63967 CQ7S3X 46837648 IC50 = 1300 nM T63967 CL7VN1 46837649 IC50 = 12000 nM T63967 CU7OG4 46837651 IC50 = 10000 nM T63967 C5WNL1 46837652 IC50 = 4800 nM T63967 COX2H5 46837653 IC50 = 12000 nM T63967 CWZY17 46837780 IC50 = 9200 nM T63967 CV2NT3 46837781 IC50 = 12000 nM T63967 CT83MU 46837782 IC50 = 27000 nM T63967 C5TY3Q 46837783 IC50 = 1800 nM T63967 CWJF83 46837784 IC50 = 12000 nM T63967 C0ZSY5 46837785 IC50 = 6300 nM T63967 CBQJ74 46837922 IC50 = 14000 nM T63967 C8UWQ2 46837923 IC50 = 7500 nM T63967 CCX8T0 46837924 IC50 = 7100 nM T63967 CBH49N 46837925 IC50 = 42000 nM T63967 CE71GL 46846404 Ki > 1000 nM T63967 CQ8KI6 46878168 EC50 = 320 nM T63967 CK9NM5 46935872 Ki = 8000 nM T63967 C5G7QD 47461992 IC50 = 70100 nM T63967 CY7O6D 49780138 EC50 = 400 nM T63967 C7U5LR 49780139 IC50 > 100000 nM T63967 CXI69G 49780140 IC50 = 3900 nM T63967 CRU36C 49780141 IC50 > 100000 nM T63967 C7E3JM 49780142 IC50 = 780 nM T63967 CBY2T0 49780345 IC50 = 250 nM T63967 CXC5S7 49780346 EC50 = 10 nM T63967 CY3H2U 49780347 EC50 = 220 nM T63967 CKJ1V7 49780348 IC50 = 16300 nM T63967 C67GSN 49780349 EC50 = 1220 nM T63967 C08JRU 49780550 EC50 = 760 nM T63967 CMB3I2 49780552 IC50 = 19900 nM T63967 CH93YJ 49780554 EC50 = 1140 nM T63967 C3XEF8 49780556 IC50 = 3820 nM T63967 CR0XM7 49780558 IC50 = 14100 nM T63967 CXAW34 49780561 IC50 = 21000 nM T63967 CQF5Z0 49783448 Ki = 2000 nM T63967 C2AWC6 49783449 Ki = 900 nM T63967 CP8E4O 49788655 IC50 = 112 nM T63967 CMI0J4 49788727 IC50 = 31.4 nM T63967 CU8O9W 49788729 IC50 = 25.8 nM T63967 C9QH1W 49788731 IC50 = 14.6 nM T63967 C2UO0F 49799236 IC50 > 100000 nM T63967 C6FH8G 49799237 IC50 > 100000 nM T63967 CZ76MQ 49799633 IC50 = 20000 nM T63967 CU28RO 49799634 IC50 = 11000 nM T63967 CN89XG 49799642 IC50 = 9000 nM T63967 C85MBT 49799643 IC50 = 6500 nM T63967 CZJV13 49852019 IC50 = 1800 nM T63967 CSL8M9 49852020 IC50 = 16000 nM T63967 CWCY74 49852021 IC50 = 7700 nM T63967 CI08OL 49852022 IC50 = 14000 nM T63967 C1BH4A 49852023 IC50 = 29000 nM T63967 C5TH3U 49859909 EC50 = 85000 nM T63967 CR53VH 49862169 Ki > 832 nM T63967 C8WRF4 49862171 Ki > 614 nM T63967 C5N4VK 49862173 Ki = 477 nM T63967 CX94UB 49862175 Ki > 309 nM T63967 C15OJH 49862213 Ki > 419 nM T63967 CT3WH4 49862215 Ki = 252 nM T63967 C15JDC 49862217 Ki = 149 nM T63967 CC97JM 49862219 Ki = 1860 nM T63967 CT39UZ 49862259 Ki > 1503 nM T63967 CTYH68 49862261 Ki > 1040 nM T63967 CHBT02 49862263 Ki > 575 nM T63967 C47WAJ 49862265 Ki = 250 nM T63967 CV96ZG 49862267 Ki = 336 nM T63967 CQ38SD 49862303 Ki = 2905 nM T63967 CL7KG5 49862305 Ki > 604 nM T63967 C9G7LW 49862307 Ki = 745 nM T63967 CGI23Z 49862361 Ki > 615.5 nM T63967 CAI26L 49862363 Ki > 962.5 nM T63967 C2RY0J 50878551 Ki > 10000 nM T63967 CL2P8X 52920232 EC50 > 100000 nM T63967 C42ROG 52920234 EC50 > 100000 nM T63967 CCP0V7 52920236 EC50 > 100000 nM T63967 CU2WT8 52941697 IC50 = 2.58 nM T63967 C64WKB 53242105 Ki = 1.7 nM T63967 C1VMW6 53242107 Ki = 1 nM T63967 CU97LK 53242130 Ki = 130 nM T63967 CEK6X4 53242144 Ki = 3 nM T63967 C23VPH 53242146 Ki = 150 nM T63967 C5R4PV 53245679 Ki > 31622.78 nM T63967 C3AKS2 53302872 Ki = 476 nM T63967 C6A7VE 53414666 Ki = 200 nM T63967 CUF61N 53706656 Ki = 0.95 nM T63967 CEY2B8 54583277 IC50 = 7200 nM T63967 C6ME0B 54584239 IC50 = 12000 nM T63967 CE7WZ8 54754345 EC50 = 10000 nM T63967 C7E9TR 56589586 EC50 = 100 nM T63967 C8DO6C 56594103 EC50 = 512.86 nM T63967 C6QHA3 56594105 EC50 = 72443.6 nM T63967 CVHC26 56594107 EC50 = 3548.13 nM T63967 CID40G 56594247 EC50 = 6770 nM T63967 C7AM2S 56594249 EC50 = 1220 nM T63967 CQO86Z 56594251 EC50 = 16595.87 nM T63967 CGP37R 56594253 EC50 = 18620.87 nM T63967 CNP6K0 56594255 EC50 = 3981.07 nM T63967 CP5R4Y 56595310 EC50 = 36 nM T63967 C8SZ5T 56595439 IC50 = 16 nM T63967 C9VQ7T 56595564 IC50 = 44 nM T63967 CQ71VT 56643499 EC50 = 300 nM T63967 C4O6ID 56666906 EC50 = 10000 nM T63967 CPO8M4 56675778 EC50 = 320 nM T63967 C7L2JC 56680506 EC50 = 10000 nM T63967 C3H1PQ 56835059 IC50 = 6600 nM T63967 C6V5XD 56926498 IC50 > 100000 nM T63967 C8BOP0 56926617 IC50 > 100000 nM T63967 C94PJS 56926722 IC50 > 100000 nM T63967 C06NVX 56926723 IC50 = 83000 nM T63967 CQ0GH2 56926724 IC50 = 12200 nM T63967 C1TEQ0 56926725 IC50 = 20900 nM T63967 C7H6WK 56951366 EC50 = 34.6 nM T63967 CZHE92 56951368 EC50 = 15.7 nM T63967 CR2N7Z 56951370 EC50 = 18.2 nM T63967 C9V3CZ 56951372 IC50 = 19.6 nM T63967 C4OXY0 56951374 EC50 = 44.4 nM T63967 CFVE45 56951376 EC50 = 48.9 nM T63967 C0C4JD 56951495 IC50 = 5.6 nM T63967 CS9KA0 56951497 EC50 = 43.1 nM T63967 CEG4N8 57334716 EC50 > 100000 nM T63967 CT75BQ 57390841 IC50 = 5900 nM T63967 C20KGJ 57390893 IC50 = 14454.4 nM T63967 C76VTP 57390894 IC50 = 7079.46 nM T63967 C5CG8V 57390895 IC50 = 6456.54 nM T63967 CNB85W 57391663 Ki > 31622.78 nM T63967 CCVI85 57391664 Ki > 31622.78 nM T63967 CX48RS 57391706 Ki > 31622.78 nM T63967 CID85U 57392658 IC50 = 5600 nM T63967 C63HMW 57393442 Ki > 31622.78 nM T63967 CC7R8I 57394370 IC50 = 25100 nM T63967 CLH9Z5 57394409 IC50 = 11481.54 nM T63967 C8J4FQ 57396124 IC50 = 4168.69 nM T63967 C83BUR 57396127 IC50 = 6500 nM T63967 CK4F0Z 57396175 IC50 = 19952.62 nM T63967 C4WDS2 57396902 Ki > 31622.78 nM T63967 CPO50Z 57397665 Ki > 31622.78 nM T63967 CBJ4O8 57397943 IC50 = 8128.31 nM T63967 C0QRL3 57397986 IC50 = 10232.93 nM T63967 CO75FJ 57397988 IC50 = 11748.98 nM T63967 C0PCS9 57398597 Ki > 31622.78 nM T63967 C3YVT8 57398685 Ki > 31622.78 nM T63967 CUN0R4 57399583 IC50 = 12589.25 nM T63967 C40FXL 57399584 IC50 = 3900 nM T63967 C2DTL4 57399630 IC50 = 2398.83 nM T63967 CTEP10 57399631 IC50 = 4265.8 nM T63967 CO2MZ8 57399632 IC50 = 2818.38 nM T63967 C93UHT 57399633 IC50 = 9549.93 nM T63967 CU8JW6 57399634 IC50 = 20892.96 nM T63967 CA1LW2 57400332 Ki > 31622.78 nM T63967 C9UMV6 57401339 IC50 = 2884.03 nM T63967 C1WHQ4 57401340 IC50 = 4300 nM T63967 C83MZY 57401393 IC50 = 6918.31 nM T63967 CX4T1A 57403094 IC50 = 17782.79 nM T63967 CSZL18 57403141 IC50 = 10000 nM T63967 C9UQF0 57403142 IC50 = 14454.4 nM T63967 C8PHB9 57403143 IC50 = 9120.11 nM T63967 C9K4SR 57403146 IC50 = 16595.87 nM T63967 CV31DZ 57485530 Ki = 0.2 nM T63967 CZ4G2Y 57485620 Ki = 0.2 nM T63967 C9G5JE 57485797 Ki = 0.26 nM T63967 CR2V6D 57485798 Ki = 0.8 nM T63967 CG1TP6 57485799 Ki = 0.7 nM T63967 CON1Z4 57485800 Ki = 0.3 nM T63967 CDW7N1 57486266 Ki = 0.4 nM T63967 CCM98N 57486336 Ki = 0.4 nM T63967 CV2J9A 57663655 IC50 = 7943.28 nM T63967 COT69D 58081856 EC50 > 100000 nM T63967 CE8V0W 58081870 EC50 > 100000 nM T63967 C9V8HI 58088056 EC50 > 100000 nM T63967 CMY5N3 58088118 EC50 > 100000 nM T63967 CP15TC 58201402 Ki = 5.2 nM T63967 CW03VZ 58201405 Ki = 5 nM T63967 CP47JL 58201407 Ki = 17 nM T63967 CMKN28 58201409 Ki = 1 nM T63967 CP8G5N 58201418 Ki = 30 nM T63967 C0TML6 58201419 Ki = 1.4 nM T63967 CB32IW 58201420 Ki = 9 nM T63967 CRC51J 58201424 Ki = 7.3 nM T63967 C2XCI7 58312740 Ki = 200 nM T63967 C3KJ7N 58488107 Ki = 4 nM T63967 COQ52A 59268918 Ki = 5 nM T63967 C4S7VM 59268924 Ki = 39 nM T63967 CYV48O 59268925 Ki = 8 nM T63967 C4N2FX 59268932 Ki = 3 nM T63967 CSW42A 59268935 Ki = 50 nM T63967 CVN48B 59268936 Ki = 11 nM T63967 CYSC50 59268939 Ki = 3 nM T63967 CTR7E8 59268940 Ki = 23 nM T63967 CHR48L 59268945 Ki = 8 nM T63967 C1TJ6W 59268948 Ki = 32 nM T63967 C3EJ6I 59268964 Ki = 16 nM T63967 CT61RD 59268965 Ki = 22 nM T63967 C9OS6X 59361675 Ki = 30 nM T63967 C1J5PV 59361705 Ki = 24 nM T63967 C68WRJ 59403312 Ki = 180 nM T63967 C6OJH7 59403341 Ki = 13 nM T63967 CX90RF 66211794 Ki = 250 nM T63967 CXN68J 66212381 Ki = 490 nM T63967 CXR63E 66212976 Ki = 23 nM T63967 C65UFK 66213161 Ki = 26 nM T63967 C9BF6L 66797369 IC50 = 58 nM T63967 C4S0IK 67144490 Ki = 700 nM T63967 CYB8S7 67235023 Ki = 6 nM T63967 CRSX31 68024489 Ki = 8 nM T63967 CPA38K 68024616 Ki = 13 nM T63967 CGU14E 68024620 Ki = 33 nM T63967 C38FDK 68024820 Ki = 53 nM T63967 CR0Q4N 68465506 Ki = 0.5 nM T63967 C5Q1PF 68611040 IC50 = 10.2 nM T63967 CF9TX0 69604735 Ki = 21 nM T63967 CZNQ13 69920709 Ki = 1.1 nM T63967 CA54SE 69920710 Ki = 5.4 nM T63967 CUL2R9 69920740 Ki = 17 nM T63967 CE0N4K 70675110 Ki = 515 nM T63967 C3CB0P 70701321 EC50 = 1200 nM T63967 C4VIB5 71099540 Ki = 5.9 nM T63967 CIE9A8 71099590 Ki = 53 nM T63967 C0DX3I 71449982 Ki = 1158 nM T63967 C5BH6L 71450029 Ki = 9.6 nM T63967 CQE53F 71450030 Ki = 0.9 nM T63967 CY5XZ3 71450042 EC50 = 38 nM T63967 C96JMX 71450130 Ki = 9 nM T63967 CZCT16 71450152 Ki = 1200 nM T63967 C4W9AV 71450153 Ki = 2300 nM T63967 C60AXY 71450154 Ki = 400 nM T63967 CQ1G5M 71450155 Ki = 500 nM T63967 C1HN0O 71450156 Ki = 1600 nM T63967 CS3N9F 71450157 Ki = 3300 nM T63967 CV9CO0 71450158 Ki = 400 nM T63967 CY8SG1 71450159 Ki = 1500 nM T63967 C2I4CF 71450171 Ki = 1 nM T63967 CRX2E6 71451808 Ki = 22 nM T63967 CQ5XI6 71451809 Ki = 105 nM T63967 C9J0NM 71451810 Ki = 0.2 nM T63967 C5SX4G 71451811 Ki = 2.2 nM T63967 CZ42AI 71451812 Ki = 0.2 nM T63967 CB6V1U 71451813 Ki = 0.4 nM T63967 C9DH7V 71451944 Ki = 19 nM T63967 CL2A9E 71451983 Ki = 2100 nM T63967 C2BGU6 71451984 Ki = 1500 nM T63967 CA69ND 71451985 Ki = 2100 nM T63967 CADC24 71451986 Ki = 500 nM T63967 CJ01HW 71451994 Ki = 7 nM T63967 C7AFY5 71452017 Ki = 980 nM T63967 C70RFX 71452018 Ki = 760 nM T63967 CI8YM0 71453627 Ki = 0.6 nM T63967 C1OS8W 71453628 Ki = 2.8 nM T63967 C89KME 71453629 Ki = 0.7 nM T63967 CDGO46 71453630 Ki = 0.3 nM T63967 C3UW8E 71453631 Ki = 9.4 nM T63967 C91CNU 71453666 Ki = 0.9 nM T63967 C7EU0L 71453717 EC50 = 35 nM T63967 C3EBR5 71453718 IC50 > 100 nM T63967 CV0Q4C 71453769 Ki = 27 nM T63967 CJL26M 71453770 Ki = 45 nM T63967 CJ1RO8 71453794 Ki = 1400 nM T63967 C7JGE0 71453795 Ki = 900 nM T63967 CQ0W3F 71453796 Ki = 4400 nM T63967 CE7U4Q 71453797 Ki = 200 nM T63967 C2HS8T 71453798 Ki = 830 nM T63967 CKHF18 71453822 Ki = 1500 nM T63967 CI8RM2 71453823 Ki = 5100 nM T63967 CTLV67 71455343 EC50 = 19.1 nM T63967 CE96BS 71455355 Ki = 1 nM T63967 CLX57K 71455356 Ki = 2.1 nM T63967 CNGK53 71455357 Ki = 0.6 nM T63967 C8N4IJ 71455358 Ki = 1.7 nM T63967 CDC54A 71455359 Ki = 13 nM T63967 CQMZ91 71455409 EC50 = 95 nM T63967 C4SRA8 71455410 EC50 = 66 nM T63967 CYJT51 71455446 EC50 > 100 nM T63967 C5MFX7 71455447 IC50 = 32 nM T63967 C8Z4ES 71455499 Ki = 60 nM T63967 CFOH06 71455500 Ki = 16 nM T63967 CT79WZ 71455501 Ki = 5 nM T63967 CC1J7O 71455527 Ki = 1600 nM T63967 CSK73V 71455528 Ki = 600 nM T63967 CSI8C3 71455529 Ki > 5000 nM T63967 C71PCM 71455535 Ki = 13 nM T63967 CSR6I8 71455553 Ki = 400 nM T63967 CN31FI 71455554 Ki = 1300 nM T63967 CFMS41 71457131 Ki = 56 nM T63967 C18UJA 71457132 Ki = 3418 nM T63967 CO5B7Z 71457133 Ki = 0.4 nM T63967 CK10DR 71457134 Ki = 0.1 nM T63967 CCFH76 71457135 Ki = 1.3 nM T63967 CY4U7W 71457136 Ki = 0.3 nM T63967 CYA78X 71457185 EC50 > 100 nM T63967 C0Y4UB 71457186 EC50 > 100 nM T63967 CH84SU 71457187 EC50 = 28 nM T63967 CDQ91P 71457319 Ki = 500 nM T63967 CS8ZC6 71457320 Ki = 500 nM T63967 CY54OR 71457321 Ki = 1500 nM T63967 CO5Z7A 71457322 Ki = 140 nM T63967 CZDF62 71457323 Ki = 1600 nM T63967 CFW9G2 71457348 Ki = 740 nM T63967 CGYS73 71457349 Ki = 1000 nM T63967 CS8Q5A 71457513 Ki = 2220 nM T63967 CN0AH1 71458995 Ki = 0.4 nM T63967 C7V0CY 71458996 Ki = 797 nM T63967 CH7U6N 71458997 Ki = 0.7 nM T63967 CUC0T8 71458998 Ki = 0.2 nM T63967 C96NIY 71459035 Ki = 0.3 nM T63967 C1WME8 71459126 Ki = 12 nM T63967 C0HTE9 71459151 Ki = 900 nM T63967 C3IJ1A 71459152 Ki = 900 nM T63967 C5IAT7 71459153 Ki = 200 nM T63967 C4S9BP 71459154 Ki = 900 nM T63967 CP1M7A 71459155 Ki = 1000 nM T63967 CB4M3E 71459156 Ki = 200 nM T63967 C3B7PW 71459157 Ki = 900 nM T63967 C8IVG6 71459158 Ki = 1200 nM T63967 CH9QF6 71459203 Ki = 1300 nM T63967 CW2YF0 71459204 Ki = 330 nM T63967 C0O8LQ 71460785 EC50 = 8.8 nM T63967 CU5D0T 71460792 Ki = 18 nM T63967 CW58SI 71460793 Ki = 0.3 nM T63967 CU7CZ6 71460794 Ki = 24 nM T63967 CZKD91 71460795 Ki = 4.4 nM T63967 CWJ1I2 71460832 Ki = 0.6 nM T63967 C0G4SZ 71460833 Ki = 1 nM T63967 C5TSZ4 71460834 Ki = 1.4 nM T63967 C2C1JW 71460847 EC50 > 100 nM T63967 CUXK17 71460848 EC50 = 97.72 nM T63967 CKM9O5 71460849 EC50 > 100 nM T63967 CWE61H 71460892 EC50 = 53.7 nM T63967 C69UGX 71460958 Ki = 1100 nM T63967 CH57RZ 71460959 Ki = 3600 nM T63967 C1UP7D 71460960 Ki = 1000 nM T63967 COH7P4 71460982 Ki = 620 nM T63967 CZO67H 71460983 Ki = 1300 nM T63967 C7AQS1 71460984 Ki = 1100 nM T63967 CV37ZJ 71462520 Ki = 1.9 nM T63967 C86IYC 71462521 Ki = 85 nM T63967 CFD1B9 71462522 Ki = 1.1 nM T63967 C3YZ6W 71462523 Ki = 3 nM T63967 CK3N6Z 71462524 Ki = 0.4 nM T63967 CX6V7B 71462553 EC50 > 100 nM T63967 CUP15I 71462588 EC50 > 100 nM T63967 C1MKL2 71462677 Ki = 1200 nM T63967 C2EU1R 71462678 Ki = 500 nM T63967 CU93PT 71462679 Ki = 600 nM T63967 CLS59K 71462680 Ki = 1400 nM T63967 C1V0ZI 71462681 Ki = 500 nM T63967 C6D0TN 71462682 Ki = 2300 nM T63967 CZW76V 71462683 Ki = 600 nM T63967 CM0HG2 71462689 Ki = 15 nM T63967 CG7ZE8 71462717 Ki = 9000 nM T63967 CXL03K 71522989 Ki = 0.049 nM T63967 CW05MP 71525308 EC50 = 310 nM T63967 CW1O3S 71569952 Ki = 1.2 nM T63967 CV5CO4 71569953 Ki = 0.076 nM T63967 CB3P9N 71569954 Ki = 0.093 nM T63967 CYL4J9 71569955 Ki = 0.083 nM T63967 CH53RK 71569956 Ki = 0.032 nM T63967 CW64OJ 71569957 Ki = 0.043 nM T63967 C7HZ3E 71569958 Ki = 0.031 nM T63967 C0C5VM 71569959 Ki = 0.05 nM T63967 C4PKN7 71570101 Ki = 0.072 nM T63967 CAOQ74 71570102 Ki = 0.046 nM T63967 C45VNU 71570103 Ki = 0.26 nM T63967 C7MI1U 71584798 IC50 = 130 nM T63967 C2VYX9 71584824 IC50 = 51 nM T63967 C50HXU 71584826 IC50 = 260 nM T63967 C3HN5E 71584828 EC50 = 160 nM T63967 CE05IZ 71584829 IC50 = 1600 nM T63967 CJ7ER8 71682669 Ki = 18 nM T63967 C05CTI 71682670 Ki = 1 nM T63967 CMKP08 71682671 Ki = 4 nM T63967 CT34ZA 71682672 Ki = 43 nM T63967 C5BO6T 71682826 Ki = 43 nM T63967 CE50MN 71682827 Ki = 110 nM T63967 CAG7D4 71682974 Ki = 1.9 nM T63967 C9C3EG 71682975 Ki = 6 nM T63967 C20NXV 71682976 Ki = 23 nM T63967 CAE0L6 71716729 EC50 = 19000 nM T63967 C7W1RU 71727769 IC50 > 100000 nM T63967 CQJ70U 71727770 IC50 = 20500 nM T63967 C35IOD 71727771 IC50 = 80700 nM T63967 CCF6M0 71727772 IC50 > 100000 nM T63967 CMT9S5 71727773 IC50 = 23200 nM T63967 CI01GP 71727774 IC50 = 37600 nM T63967 C52MJY 71727775 IC50 = 15400 nM T63967 C3NK1F 71727895 IC50 = 54100 nM T63967 CW72HR 71727896 IC50 > 100000 nM T63967 C7INR8 71727897 IC50 > 100000 nM T63967 CJZ5K9 71727898 IC50 > 100000 nM T63967 CJYM35 71727899 IC50 > 100000 nM T63967 CQ24PX 71727900 IC50 > 100000 nM T63967 C08YLD 71727901 IC50 > 100000 nM T63967 C17IXA 71728020 IC50 > 100000 nM T63967 C6F3NV 71728021 IC50 > 100000 nM T63967 C3FZ8C 71728022 IC50 > 100000 nM T63967 C8OGQ1 71728023 IC50 > 100000 nM T63967 CE1Z0Y 71728024 IC50 = 14800 nM T63967 CO4G6R 71728025 IC50 = 22400 nM T63967 CY6I5V 71746415 EC50 = 23 nM T63967 C7N6ZF 71746417 EC50 = 14.4 nM T63967 CD83PF 71746602 EC50 = 6.2 nM T63967 CHW18L 72703052 Ki = 477 nM T63967 C6NOM3 72703256 Ki = 562 nM T63967 C0GQ7F 72703471 Ki = 885 nM T63967 CMZ19D 72703472 Ki = 141 nM T63967 CCE9W7 72703473 Ki = 4000 nM T63967 CDNY35 72712462 Ki > 100000 nM T63967 CYN0X1 72712463 Ki > 1000 nM T63967 CWVI40 72712464 Ki = 0.11 nM T63967 C1KT0W 73347339 Ki = 217 nM T63967 C87TLQ 73347340 Ki = 22.4 nM T63967 CY56RE 73347561 Ki = 2.9 nM T63967 CD8OT4 73348844 Ki = 11.2 nM T63967 CL73CV 73350432 Ki = 1.2 nM T63967 CEBL05 73350433 Ki = 15.5 nM T63967 C71LER 73350667 Ki = 0.2 nM T63967 CP62JM 73350668 Ki = 20 nM T63967 C5ILK3 73351944 Ki = 23.4 nM T63967 CER79N 73352166 Ki = 28 nM T63967 CIX69R 73353186 IC50 = 5 nM T63967 CL6S2I 73353403 Ki = 151 nM T63967 CGD3K1 73354915 Ki = 8.1 nM T63967 CYL5C0 73355120 Ki = 1 nM T63967 C5PJ4Z 73356479 Ki = 460 nM T63967 CZY29O 73356690 Ki = 2400 nM T63967 CKD42Z 75113427 Ki = 0.35 nM T63967 CIFM07 75582810 Ki = 3.5 nM T63967 C3V9FS 75582871 Ki = 0.5 nM T63967 C1BA3C 76311214 Ki = 600 nM T63967 CT0N4Q 76311216 IC50 = 3900 nM T63967 CYM3V2 76312105 Ki = 11200 nM T63967 CWG93E 76314835 IC50 = 4200 nM T63967 CFG3N4 76318436 IC50 = 14800 nM T63967 C72USC 76322102 Ki = 1600 nM T63967 CQ4D8U 76325731 IC50 > 100000 nM T63967 C7MOY0 76326531 Ki = 734 nM T63967 CU89CH 76328290 IC50 = 309 nM T63967 C6S9CQ 76329290 IC50 = 9500 nM T63967 CZ4I0Y 76330174 Ki = 4 nM T63967 C5YE3Q 76332941 IC50 = 9100 nM T63967 CKZ19D 76336550 IC50 = 4400 nM T63967 CJ9N1O 76336552 IC50 = 20000 nM T63967 COZ70Q 77430458 Ki = 2800 nM T63967 CPHO43 77907039 Ki = 449 nM T63967 COFC93 84076119 Ki = 320 nM T63967 CZ1KQ4 89273585 Ki = 51 nM T63967 CH3PY1 89273597 Ki = 160 nM T63967 CZEW07 89273598 Ki = 16 nM T63967 C3S4XB 89273612 Ki = 14 nM T63967 CB02MN 89273615 Ki = 3.9 nM T63967 C9XP6Q 89273626 Ki = 22 nM T63967 C4Q7OM 89273629 Ki = 7 nM T63967 CXT72M 89273630 Ki = 1 nM T63967 CZCV56 89943572 Ki = 10436 nM T63967 CKI70A 89943585 Ki = 1000 nM T63967 CE6R1X 89943698 Ki > 1000 nM T63967 CUX53L 89943718 Ki = 5201 nM T63967 CEI2S7 89943719 Ki = 748 nM T63967 C3EKN1 89943828 Ki = 1000 nM T63967 C8ASH6 89943878 Ki > 1000 nM T63967 CH21GZ 89943908 Ki = 1000 nM T63967 CFI10Y 118716172 EC50 = 12 nM T63967 CJ40LN 118721306 IC50 = 10 nM T63967 C7ZJO9 118721308 EC50 > 1000 nM T63967 CO32DI 118721309 EC50 = 15.85 nM T63967 CL67KA 118721311 IC50 = 19.95 nM T63967 C1KI3L 118721314 IC50 = 12.59 nM T63967 C2TO8V 122185335 EC50 = 4400 nM T63967 CDQO08 122185338 EC50 = 73000 nM T63967 CXVF35 122185349 EC50 = 13 nM T63967 CAHY43 122188151 IC50 = 90 nM T63967 C2MYB7 122188152 IC50 = 300 nM T63967 C25WZN 122188153 IC50 = 200 nM T63967 CE0VY6 122188155 IC50 = 800 nM T63967 CY6O8L 122188157 IC50 = 100 nM T63967 CCK1L8 122553340 Ki = 750 nM T63967 CR0P7N 122553341 Ki = 627 nM T63967 CKDM68 123133764 EC50 > 25000 nM T63967 C93OKB 124089453 EC50 = 275 nM T63967 CRT3H8 134130624 EC50 > 1000 nM T63967 COQ83N 134131946 EC50 > 1000 nM T63967 CY0K3C 134133420 EC50 = 16.98 nM T63967 CWJ71I 134134377 EC50 > 1000 nM T63967 C1N7EU 134140902 EC50 = 125 nM T63967 C5UR7T 134147102 EC50 = 15.85 nM T63967 C7X2QN 134153793 EC50 = 30.9 nM T63967 C1GY2T 135156251 EC50 > 10000 nM T63967 CKZ59F 135412796 Ki = 340 nM T63967 CLE38V 135508231 Ki = 19 nM T63967 CX0LF6 137633214 EC50 > 100000 nM T63967 C93ZPK 137635141 EC50 > 100000 nM T63967 COI42G 137635637 Ki = 9700 nM T63967 CTU9Y7 137635902 EC50 > 100000 nM T63967 CN8Y4B 137637992 IC50 = 51000 nM T63967 C3UT9L 137643408 EC50 > 100000 nM T63967 CVJ0Q7 137644763 EC50 > 100000 nM T63967 C9K7VP 137644928 EC50 > 100000 nM T63967 CQ5H2Y 137645815 EC50 > 100000 nM T63967 CV9T6B 137647317 EC50 > 100000 nM T63967 C3Y2SW 137649484 EC50 > 100000 nM T63967 C6RJ8V 137649905 EC50 > 100000 nM T63967 CCY0D8 137652873 EC50 = 10100 nM T63967 CVON14 137654242 EC50 > 100000 nM T63967 CJC95L 137654434 EC50 > 100000 nM T63967 COVD20 137655697 EC50 > 100000 nM T63967 C6CYW8 137657023 EC50 > 100000 nM T63967 CS3K4D 137659736 EC50 > 100000 nM T63967 CX39HQ 137659815 EC50 > 100000 nM T63967 C4GOE0 137660090 EC50 > 100000 nM T63967 CP48RG 137660174 EC50 > 100000 nM T63967 C0B6HQ 137660214 EC50 > 100000 nM T63967 C3FZL5 141725921 EC50 = 6140 nM T63967 C43URC 145954515 EC50 > 10000 nM T63967 COY76F 145972407 EC50 = 1900 nM T63967 CG9QD6 145980121 Ki > 3000 nM T63967 C3U0HD 145986545 Ki > 3000 nM T63967 C7XB0C 145989786 Ki = 0.27 nM T63967 C9U4IN 145989794 Ki > 3000 nM T63967 C8V6DI 145990201 Ki > 3000 nM T63967 CMY8S3 145991947 Ki > 3000 nM T63967 C6Q3XK 146680925 Ki = 6392 nM T63967 C6DCN9 146680926 Ki = 519 nM T63967 C9F6LV 155512339 Ki = 1962 nM T63967 CM7DV8 155514108 IC50 = 25.6 nM T63967 CT64LK 155514460 Ki = 1980 nM T63967 C5AS9Y 155515572 EC50 = 1000 nM T63967 CMV2G7 155515603 Ki = 537 nM T63967 C7DBH6 155516230 Ki = 1262 nM T63967 CW8IV5 155516492 IC50 = 28.2 nM T63967 C5GAS9 155521191 Ki = 414 nM T63967 CHC38D 155522533 Ki = 3894 nM T63967 CK01QX 155522758 Ki = 461 nM T63967 C19POZ 155523848 IC50 = 21.4 nM T63967 C5U6IO 155527752 EC50 = 520 nM T63967 CFAY97 155528499 IC50 = 6700 nM T63967 C2YXJ9 155529181 IC50 = 12.1 nM T63967 C57HKR 155529699 IC50 = 5.43 nM T63967 CLYV89 155530137 Ki = 5059 nM T63967 C3VOB7 155532967 Ki = 9010 nM T63967 CO07HD 155533348 Ki = 668 nM T63967 CMK0U4 155537399 Ki = 7050 nM T63967 C8Y4PI 155541561 IC50 = 47.4 nM T63967 CD3EW6 155546334 IC50 = 44.3 nM T63967 C7W5ZC 155547147 EC50 = 600 nM T63967 CM50TS 155547626 Ki = 7389 nM T63967 CROV92 155554398 Ki = 1013 nM T63967 C6RU4P 155557819 IC50 = 20.8 nM T63967 CW51RT 155564442 IC50 = 22.5 nM T63967 CR24FZ 155568280 Ki = 35300 nM T63967 CO0U9B 11587705 Ki = 29 nM T63967 CB0LH8 11602721 IC50 = 1995.26 nM T63967 CTAK49 11660066 IC50 = 5011.87 nM T63967 C7NWZ6 442202 IC50 = 970 nM T63967 CUZ1D8 44564663 IC50 = 10000 nM T63967 D00GDI 45487890 IC50 = 29 nM T63967 D00QCP 46837647 IC50 = 6400 nM T63967 D00WPU 11983356 Ki = 0.062 nM T63967 D01OMG 11998180 EC50 = 990 nM T63967 D01YED 45141808 IC50 = 57 nM T63967 D02LWF 44274422 IC50 = 1.1 nM T63967 D02ZIQ 43227131 IC50 = 30 nM T63967 D03FEV 9793858 Ki = 35 nM T63967 D03JPN 11173546 Ki > 100000 nM T63967 D03SYO 15860335 Ki = 58 nM T63967 D03YQY 46837650 IC50 = 6000 nM T63967 D04HQP 44366245 Ki = 510 nM T63967 D04KZX 44542809 IC50 = 10 nM T63967 D05PLF 3031066 IC50 = 33 nM T63967 D05ZUX 44207909 Ki >= 1000 nM T63967 D06FLU 10480509 Ki = 31000 nM T63967 D06KYM 44302712 Ki = 28 nM T63967 D06LCK 45141805 IC50 = 71 nM T63967 D08SCF 159548 IC50 = 80.2 nM T63967 D09BSE 10409038 Ki = 30000 nM T63967 D09BYB 45487941 IC50 = 17 nM T63967 D09XWL 45141379 IC50 = 81 nM T63967 D0A7HM 10197862 Ki = 21 nM T63967 D0C0GL 3031062 IC50 = 15 nM T63967 D0G0CJ 45141380 IC50 = 42 nM T63967 D0G1XP 44543273 IC50 = 9.8 nM T63967 D0GY8R 45141807 IC50 = 56 nM T63967 D0H4AD 44542509 IC50 = 23 nM T63967 D0J5EF 215051 IC50 = 21 nM T63967 D0LH4L 10154 Ki = 3000 nM T63967 D0O2LC 44543272 IC50 > 100 nM T63967 D0P2HR 3510 Ki = 38000 nM T63967 D0P9ED 11601009 Ki = 0.038 nM T63967 D0P9EO 45141381 IC50 = 25 nM T63967 D0Q8IQ 43794735 IC50 > 100 nM T63967 D0R4RN 1204 EC50 = 0.0088 nM T63967 D0R8EV 3027752 IC50 = 8.6 nM T63967 D0R8YJ 44366246 Ki = 1770 nM T63967 D0T2RY 9948320 Ki >= 1000 nM T63967 D0T9SK 6380 Ki = 24 nM T63967 D0U2HZ 9816611 Ki = 256 nM T63967 D0U3SB 45141806 IC50 = 74 nM T63967 D0UH8F 44274190 IC50 = 8 nM T63967 D0UX5M 7330459 Ki = 540 nM T63967 D0V0AW 9823180 Ki = 12 nM T63967 D0V2KB 44423690 Ki = 970 nM T63967 D0V7HJ 9794401 Ki = 0.5 nM T63967 D0VY9K 45141809 IC50 > 100 nM T63967 D0X7CX 31762 IC50 = 20 nM T63967 D0XY9E 3029724 IC50 = 7.7 nM T63967 D0Y7CS 44543118 IC50 = 19 nM T63967 D0ZE4C 45141608 IC50 = 31 nM T52389 D02TJS 54676038 IC50 = 5 nM T52389 D0L5MF 339455 IC50 = 45000 nM T52389 D0W0VD 3885 IC50 = 3000 nM T52389 CWI4B7 13862 IC50 = 20000 nM T52389 C7TZ3U 219751 IC50 = 105000 nM T52389 CYZ2E8 230481 IC50 = 22500 nM T52389 C1WL4K 358258 IC50 = 60000 nM T52389 C1I2YS 363151 IC50 = 45000 nM T52389 C1RT3G 372797 IC50 = 70000 nM T52389 CK6U5C 379560 IC50 = 90000 nM T52389 CVI1B6 381315 IC50 = 25000 nM T52389 C5K7DO 438560 IC50 = 1800 nM T52389 CB2GN1 438565 IC50 = 111 nM T52389 C8JC0T 438696 IC50 = 150000 nM T52389 CH7G5Y 761891 IC50 = 1470 nM T52389 CXN5K8 5320815 IC50 = 25000 nM T52389 CDF2N3 5351322 IC50 = 25000 nM T52389 CFZ50Q 5351406 IC50 = 55000 nM T52389 C90LVB 5387854 IC50 = 90000 nM T52389 CT89GA 5781276 IC50 = 250000 nM T52389 CLK6I5 14631798 IC50 = 4100 nM T52389 C5R4LE 14631799 IC50 = 8500 nM T52389 C6NYI9 22899233 IC50 = 12000 nM T52389 CIK0A7 23661722 IC50 = 2600 nM T52389 CNVD56 44420345 IC50 = 55000 nM T52389 C9YBD3 44420464 IC50 = 95000 nM T52389 CP1LJ4 44585411 IC50 = 1800 nM T52389 CTK0L3 44627376 IC50 = 2400 nM T52389 CL9NO0 44627378 IC50 = 1300 nM T52389 C9QVR3 46231191 IC50 = 188 nM T52389 C6GC7K 46231192 IC50 = 780 nM T52389 C86BIK 46231193 IC50 = 206 nM T52389 CKGV86 46231194 IC50 = 203 nM T52389 C5M1NJ 46231195 IC50 = 145 nM T52389 CIVO25 46231242 IC50 = 808 nM T52389 C5GEO9 46231243 IC50 = 92 nM T52389 CKZ83D 46231244 IC50 = 107 nM T52389 CI0F2H 46231245 IC50 = 3933 nM T52389 CY0H6O 46231246 IC50 = 3283 nM T52389 CMX69C 46231284 IC50 = 328 nM T52389 C1DJV8 46231285 IC50 = 94 nM T52389 CO74HZ 46231286 IC50 = 507 nM T52389 CJ1ME4 52941605 IC50 = 40000 nM T52389 C0SCO6 54676523 IC50 = 220 nM T52389 CZ3EO7 54676828 IC50 = 6 nM T52389 CKV63M 54677783 IC50 = 29000 nM T52389 C4VBK8 54677992 IC50 = 2300 nM T52389 CT5U7Q 54678493 IC50 = 2200 nM T52389 C57DJK 54679390 IC50 = 650 nM T52389 C7I9FJ 54679916 IC50 = 550 nM T52389 CIQH03 54680448 IC50 = 5 nM T52389 C01NIS 54680449 IC50 = 250 nM T52389 C1TRL5 54680450 IC50 = 7500 nM T52389 C9N8SK 54680452 IC50 = 21000 nM T52389 C4J7LW 54682817 IC50 = 1250 nM T52389 CCH25I 54685683 IC50 = 350 nM T52389 CH3DP1 54686240 IC50 = 8000 nM T52389 C6OC5F 54686375 IC50 = 110 nM T52389 C2LWC7 54690695 IC50 = 100 nM T52389 CG2K8L 54692153 IC50 = 200 nM T52389 CUE7A9 54694511 IC50 = 500 nM T52389 C5Z0UQ 54695479 IC50 = 44500 nM T52389 C54QHM 54695483 IC50 = 1700 nM T52389 C3GP4U 54703291 IC50 = 320 nM T52389 C0PQY7 54703981 IC50 = 5322 nM T52389 C3OU8A 54706321 IC50 = 1300 nM T52389 C8QP3G 54707106 IC50 = 920 nM T52389 CY36DA 54714086 IC50 = 18000 nM T52389 CNHF75 54714087 IC50 = 140 nM T52389 C0KVX1 54714091 IC50 = 250 nM T52389 CFB21V 54716147 IC50 = 690 nM T52389 C1K5BR 54734760 IC50 = 41000 nM T52389 C0PR2A 54736423 IC50 = 7.7 nM T52389 C14ATB 54736424 IC50 = 1150 nM T52389 C9ZX4A 54736425 IC50 = 167 nM T52389 CRG17S 54736426 IC50 = 6250 nM T52389 CA7OH0 54736427 IC50 = 4.9 nM T52389 CNA58U 54736429 IC50 = 9.9 nM T52389 CDA61P 54736430 IC50 = 0.41 nM T52389 CDH09L 54736431 IC50 = 450 nM T52389 C0AP5M 54736432 IC50 = 1497 nM T52389 C6BM2Z 54736433 IC50 = 370 nM T52389 CDS38G 54736434 IC50 = 14 nM T52389 CMJ8U9 54736435 IC50 = 96 nM T52389 C4FEX7 54736436 IC50 = 2.2 nM T52389 CL72PZ 54736437 IC50 = 2.8 nM T52389 CB36IU 54736439 IC50 = 6.3 nM T52389 CF46ER 54736440 IC50 = 6 nM T52389 CW3T7V 54736442 IC50 = 11 nM T52389 C76CRO 54736445 IC50 = 4.5 nM T52389 C6CF3N 57329528 IC50 = 6250 nM T52389 CMOV75 118727359 IC50 = 5800 nM T52389 CV68LZ 118727360 IC50 = 11000 nM T52389 CWM3K7 134149218 IC50 = 640 nM T52389 C4TUB7 134151310 IC50 = 1200 nM T52389 CD3MH9 135468602 IC50 = 73400 nM T52389 C86CQW 135493734 IC50 = 35000 nM T52389 CZUS49 135499423 IC50 = 35000 nM T52389 CP79QH 137632568 IC50 = 3100 nM T52389 C4L2CA 137641351 IC50 = 2900 nM T52389 CQ4EM8 137643157 IC50 = 3100 nM T52389 CT21CH 137659467 IC50 = 11000 nM T52389 C7W4YA 137662216 IC50 = 2400 nM T52389 C3CQ9O 145949863 IC50 = 530 nM T52389 CFN7I4 145956581 IC50 = 2040 nM T52389 C3BQY4 145957600 IC50 = 470 nM T52389 CS3O4K 145959131 IC50 = 440 nM T52389 C20IUC 145980617 IC50 = 980 nM T52389 CA81VH 145982365 IC50 = 480 nM T52389 CXS5E6 145987528 IC50 = 230 nM T52389 C30PXS 155512198 IC50 = 133900 nM T52389 CC92QZ 155516868 IC50 = 425 nM T52389 CH3E1N 155555454 IC50 = 38700 nM T52389 D00OTC 5385086 IC50 = 80000 nM T52389 D00SRM 44420298 IC50 = 2000 nM T52389 D02ONP 54736443 IC50 = 22333 nM T52389 D03CDH 54736438 IC50 = 35 nM T52389 D05GWI 83107 IC50 = 10000 nM T52389 D06BHJ 54736444 IC50 = 31 nM T52389 D07DGS 67150 IC50 = 3500 nM T52389 D07JNQ 16528 IC50 = 7500 nM T52389 D07MGN 312765 IC50 = 12500 nM T52389 D08XJX 54736428 IC50 = 39 nM T52389 D09CYJ 54711585 IC50 = 24 nM T52389 D09FMZ 54686112 IC50 = 144 nM T52389 D09ITX 54736441 IC50 = 15 nM T52389 D0A5TD 359787 IC50 = 390 nM T52389 D0AN7U 432861 IC50 = 17500 nM T52389 D0B4GV 820807 IC50 = 3250 nM T52389 D0E0DQ 371510 IC50 = 10000 nM T52389 D0E2LU 321796 IC50 = 3000 nM T52389 D0GE8S 4470790 Ki = 450 nM T52389 D0H4YP 54724899 IC50 = 14 nM T52389 D0L3VV 433916 IC50 = 2000 nM T52389 D0M0WT 264430 IC50 = 1100 nM T52389 D0O8YZ 248349 IC50 = 10000 nM T52389 D0T4RW 124496 IC50 = 700 nM T52389 D0VB8K 433914 IC50 = 3000 nM T03023 D0E3TC 44259 IC50 = 8770 nM T03023 CLS29B 46872626 IC50 > 10000 nM T03023 CV63UL 67240318 IC50 > 10000 nM T03023 COU73Y 71226944 IC50 = 19 nM T03023 C40JOZ 71235465 IC50 = 76 nM T03023 CZOD53 137633880 IC50 = 84 nM T03023 C7BJY5 137636807 IC50 = 65 nM T03023 CO89DX 137649100 IC50 = 50 nM T03023 CINE03 137652514 IC50 = 103 nM T16117 D08ZEB 2733 IC50 = 50000 nM T16117 D05QJT 9797017 IC50 = 8400 nM T16117 D07WGN 656912 Ki = 0.1 nM T16117 D0D3AI 39836 IC50 = 1600 nM T16117 D0V0NL 2146 Ki = 3300 nM T16117 D0Y7VJ 2733506 IC50 = 1500 nM T16117 CF06EN 795 Ki = 175000 nM T16117 C6N8HS 1337 Ki = 16 nM T16117 CZ0VE3 1484 IC50 = 6000 nM T16117 CFIC95 2039 Ki = 1800 nM T16117 CHM9K2 4366 IC50 = 90 nM T16117 CP62OB 5138 Ki = 14000 nM T16117 C9OF8C 5142 Ki = 160 nM T16117 C2BR0H 9221 IC50 = 178000 nM T16117 C20EWK 15347 IC50 = 1300 nM T16117 C2YN0X 18057 IC50 = 3100 nM T16117 C5TXR9 27842 IC50 = 5600 nM T16117 C0UF5P 53616 Ki = 125000 nM T16117 C9NY7L 73046 IC50 = 4300 nM T16117 CL85YU 73238 Ki = 380 nM T16117 C8CQW2 73742 IC50 = 6600 nM T16117 CZD9B8 74143 Ki = 10000 nM T16117 CIP86S 81423 IC50 > 1000000 nM T16117 CN65RF 81595 Ki = 430000 nM T16117 C6VWY5 82645 Ki = 100 nM T16117 CWI59L 88012 IC50 > 1000000 nM T16117 C0PU6F 88901 IC50 = 115000 nM T16117 CWA7P8 95894 IC50 = 100000 nM T16117 CX51OV 96652 IC50 = 158000 nM T16117 CCFW32 97525 Ki = 350000 nM T16117 C7AB0Y 107968 IC50 = 60 nM T16117 CZXU91 118425 IC50 = 2200 nM T16117 C05CIO 120987 Ki = 630 nM T16117 CP49UZ 132862 Ki = 840 nM T16117 CT7M5K 135193 IC50 = 690 nM T16117 CWG0F1 152144 IC50 = 4600 nM T16117 C56DHZ 155864 Ki = 4000 nM T16117 CW72NB 203391 Ki = 6000 nM T16117 CP18FD 203816 Ki = 14000 nM T16117 CG96BR 211124 IC50 > 50000 nM T16117 C23ABJ 262484 IC50 = 2200 nM T16117 C8B7YF 287208 IC50 > 50000 nM T16117 C3ZA0H 322632 IC50 = 50000 nM T16117 CV7K2N 322634 IC50 = 13100 nM T16117 CTK6I8 330841 IC50 = 620 nM T16117 C86SOD 351770 Ki = 1100 nM T16117 CV7PL1 410658 Ki = 800 nM T16117 C9V1WQ 415736 Ki = 14000 nM T16117 C35JRN 449021 IC50 = 35 nM T16117 C40ZOB 544920 IC50 > 50000 nM T16117 C9ABD3 656910 Ki = 0.3 nM T16117 CF7Z2I 656911 Ki = 0.15 nM T16117 C8SFX0 708870 IC50 > 50000 nM T16117 C39PAJ 764995 IC50 = 80 nM T16117 C9WNS2 867248 Ki = 125000 nM T16117 CNM06C 1375038 EC50 > 10000 nM T16117 C6U5SR 2733505 IC50 = 35000 nM T16117 CGWI36 2734673 Ki = 400 nM T16117 CWX56G 2795028 Ki = 620 nM T16117 C59BGS 2818222 Ki = 570 nM T16117 CVLT98 2843665 Ki = 32000 nM T16117 CCZ86X 2843697 Ki = 180000 nM T16117 CTF27A 2843772 Ki = 125000 nM T16117 C8K2MN 2843859 Ki = 57000 nM T16117 CH5QU8 3016310 IC50 = 2000 nM T16117 C9YW2K 3608221 Ki = 890 nM T16117 C5L7GD 3636377 Ki > 50000 nM T16117 C4VNF7 3792909 IC50 > 100000 nM T16117 CUI4F5 4247236 IC50 = 60 nM T16117 C97INL 4262401 Ki = 13000 nM T16117 C6KW9G 4469991 IC50 = 9000 nM T16117 CL7OU5 5057184 IC50 = 275000 nM T16117 CLP5G9 8775318 Ki = 140 nM T16117 CI6O2G 8775930 Ki = 290 nM T16117 C5GNH3 8776467 Ki = 170 nM T16117 C31FNY 9571038 Ki = 680 nM T16117 CC52JU 9794039 IC50 = 510 nM T16117 CVZ93W 9795163 IC50 = 380 nM T16117 CE62HS 9796600 IC50 = 220 nM T16117 C4H6JA 9797393 IC50 = 109 nM T16117 C3AWZ7 9815642 IC50 = 21700 nM T16117 C96UVG 9815901 Ki = 44000 nM T16117 CN6XG0 9816945 Ki = 190 nM T16117 CQCA72 9818336 IC50 = 58 nM T16117 CCS6E5 9819003 IC50 = 8000 nM T16117 CBC5H3 9821853 IC50 = 1150 nM T16117 CJ9KY8 9823420 IC50 = 2300 nM T16117 CX7E2G 9823715 IC50 = 36000 nM T16117 CHIO18 9834486 IC50 = 3300 nM T16117 CBZ95E 9837386 IC50 = 140 nM T16117 C8ADG2 9838603 IC50 = 75000 nM T16117 CQF37H 9839201 IC50 = 50.6 nM T16117 CP2IL5 9842658 Ki = 6.3 nM T16117 C80IET 9843967 IC50 = 140 nM T16117 CAM64J 9881505 IC50 > 100000 nM T16117 CVT64X 9891254 IC50 = 2000 nM T16117 C74UBK 9904260 IC50 = 74000 nM T16117 C0JHT5 9905692 IC50 = 250 nM T16117 CEF5Q9 9907534 IC50 = 5000 nM T16117 C85CXW 9920422 Ki = 14000 nM T16117 CBA1D9 9927237 IC50 = 120 nM T16117 C9H3PG 9927273 IC50 = 40000 nM T16117 CA05GJ 9931138 IC50 = 3500 nM T16117 C3PH5S 9931834 IC50 = 3000 nM T16117 C8P4MX 9932597 IC50 = 1040 nM T16117 C72OQJ 9942188 IC50 = 1200 nM T16117 CGU01Y 9950094 IC50 = 7800 nM T16117 C2I1JH 9950891 IC50 = 12000 nM T16117 CNB2L4 9991061 Ki = 1300 nM T16117 CG2C1Y 9994346 Ki = 350 nM T16117 CL3Y5Z 10020993 IC50 = 48 nM T16117 CYZJ64 10034809 IC50 = 36 nM T16117 C7YM4U 10060017 Ki = 410 nM T16117 CS7I1H 10068818 IC50 = 200 nM T16117 CU8RO9 10080329 Ki = 12000000 nM T16117 CTP9Z0 10084004 Ki = 540 nM T16117 C4CFP5 10084782 Ki = 460 nM T16117 C1PT8H 10085485 Ki = 2000 nM T16117 C58LCS 10103217 IC50 > 50000 nM T16117 C3GVU2 10104005 IC50 = 460 nM T16117 C9Z1HS 10149857 IC50 = 1202.26 nM T16117 CHT12V 10171540 IC50 = 18620.87 nM T16117 CD5NH1 10172593 IC50 = 13803.84 nM T16117 CJ97GV 10176386 Ki = 11 nM T16117 C7NV2T 10192988 IC50 = 26302.68 nM T16117 CHJN87 10214800 IC50 = 54 nM T16117 CHF49M 10215218 IC50 = 123026.88 nM T16117 C58KRE 10219864 IC50 = 4000 nM T16117 CK7GN4 10219896 IC50 = 70400 nM T16117 CA68IC 10220131 IC50 = 33800 nM T16117 C1FZR9 10220855 IC50 = 390 nM T16117 C3NPV0 10221335 IC50 = 790 nM T16117 CAEK83 10248425 IC50 = 42 nM T16117 C8P7WJ 10263292 IC50 = 250 nM T16117 CBP8Q2 10265375 IC50 = 200 nM T16117 CVTQ48 10286162 IC50 = 12589.25 nM T16117 CN42PW 10308710 IC50 = 8317.64 nM T16117 CS8T6Z 10313224 IC50 = 21 nM T16117 CJ3W7S 10330523 IC50 = 150000 nM T16117 C31AYP 10330543 IC50 = 170 nM T16117 CNKY10 10330544 IC50 = 100 nM T16117 C7HK2M 10332472 IC50 > 500000 nM T16117 C9P7SQ 10354581 IC50 = 50000 nM T16117 CWDA37 10358114 IC50 = 70 nM T16117 C41RXN 10376219 IC50 = 6700 nM T16117 CLZF27 10377204 Ki = 74000 nM T16117 CALW76 10398017 IC50 = 21000 nM T16117 CIHA04 10398629 Ki = 370 nM T16117 C4P8EC 10400619 IC50 = 310 nM T16117 CI0JY4 10406425 IC50 = 4400 nM T16117 CR47JC 10411355 IC50 = 500 nM T16117 C7E2VQ 10452321 IC50 = 1300 nM T16117 CG94NE 10488346 IC50 = 3300 nM T16117 CB81CA 10489359 IC50 = 6600 nM T16117 C15IWF 10496245 Ki = 40 nM T16117 CVYG70 10498721 Ki = 30400 nM T16117 C78SPQ 10499986 Ki = 150000 nM T16117 C5AFW7 10499987 Ki = 2000 nM T16117 CTN4R7 10514976 Ki = 1600 nM T16117 C2FNA0 10518871 IC50 = 82000 nM T16117 CHA40M 10521987 Ki = 170 nM T16117 C9FO8V 10523506 Ki = 10200 nM T16117 CCV50K 10523810 Ki = 370000 nM T16117 C56DVA 10524594 Ki = 8.7 nM T16117 CZ7K3C 10531193 Ki = 47000 nM T16117 C8MIC9 10537022 Ki = 1100 nM T16117 CDY6I3 10538489 Ki = 1400 nM T16117 C9CK0T 10539398 Ki = 64000 nM T16117 C8QN6S 10540046 IC50 = 26915.35 nM T16117 C1GHN4 10549183 IC50 = 140000 nM T16117 C0FTK6 10562607 Ki = 1000 nM T16117 C5FE1Z 10569061 Ki = 56 nM T16117 C7YTK5 10570902 Ki = 17000 nM T16117 C0JF6I 10575453 IC50 = 4000 nM T16117 C2X0EI 10584290 IC50 = 500 nM T16117 CCQ8P1 10585015 IC50 = 327000 nM T16117 CD68UG 10593092 IC50 = 34000 nM T16117 C1QW6P 10595933 Ki = 92000 nM T16117 CJG9L3 10607934 Ki = 340 nM T16117 C2BZ7Q 10608524 Ki = 560 nM T16117 CW4I8K 10616592 IC50 = 30000 nM T16117 C1D6GY 10630840 IC50 = 11000 nM T16117 CJD2U9 10630842 IC50 = 5900 nM T16117 CZR04I 10631254 Ki = 1000 nM T16117 C9IVH2 10631255 Ki = 800 nM T16117 C18YCZ 10632442 Ki = 450 nM T16117 CNYF76 10634991 Ki = 250 nM T16117 C7V8QW 10650502 Ki = 2400 nM T16117 CUP7V1 10651023 Ki = 7300 nM T16117 CZ7QR6 10655660 IC50 > 100000 nM T16117 C7DY3X 10656126 Ki = 3300 nM T16117 CCU7H9 10656678 Ki = 330 nM T16117 C7R3TC 10656792 IC50 = 900 nM T16117 CA95NW 10663856 Ki = 1100 nM T16117 CA4N8W 10666552 Ki = 370 nM T16117 C30FNO 10667470 Ki = 90000 nM T16117 CKG34H 10671340 Ki = 52000 nM T16117 C9R0NE 10680179 Ki = 170 nM T16117 CO03PU 10680655 IC50 = 30000 nM T16117 COWH50 10688427 Ki > 50000 nM T16117 C94OWI 10702801 IC50 = 870 nM T16117 CF84US 10704325 Ki = 1400 nM T16117 C6WC8D 10705708 Ki = 175000 nM T16117 CQUD49 10713929 Ki = 140000 nM T16117 C3EL8F 10718613 Ki = 55000 nM T16117 C4J8BY 10721117 Ki = 42 nM T16117 C89DJZ 10721313 Ki = 28400 nM T16117 C5CSV1 10727897 Ki = 660 nM T16117 C3ON1R 10736195 Ki = 300 nM T16117 C2KEY4 10753994 Ki = 1500 nM T16117 CL38ZM 10755655 Ki = 210 nM T16117 CGTX82 10761718 Ki = 11 nM T16117 CWQ23R 10766216 Ki = 110000 nM T16117 C1LM7K 10768934 Ki = 19000 nM T16117 CM2ZI5 10773629 IC50 = 2400 nM T16117 CD90OG 10776989 Ki = 570 nM T16117 COV8A4 10780100 Ki = 29000 nM T16117 C4T8XO 10786837 Ki = 2800 nM T16117 CU5WR9 10788294 Ki = 190 nM T16117 CGY24Z 10797080 IC50 = 3800 nM T16117 C8YXF1 10797487 Ki = 4800 nM T16117 CHNS51 10797903 Ki = 180 nM T16117 CDW7R0 10798324 IC50 = 1621000 nM T16117 C5CE9H 10799502 IC50 = 28000 nM T16117 CS3WY5 10799675 Ki = 4600 nM T16117 CXZ1W9 10800554 Ki = 1100 nM T16117 CV2ER7 10800919 IC50 = 500 nM T16117 CXZ82D 10807142 Ki = 2100 nM T16117 C56AMX 10810281 Ki = 330 nM T16117 C9F4GI 10822632 IC50 = 5300 nM T16117 CPJQ17 10823018 Ki = 58000 nM T16117 CHND09 10823019 Ki = 11000 nM T16117 C4O0YS 10823395 Ki = 375000 nM T16117 CL2M4B 10824083 IC50 = 24000 nM T16117 CMOE80 10825489 Ki = 700 nM T16117 CP3W2V 10830415 IC50 = 30000 nM T16117 C65FGY 10830685 IC50 = 60000 nM T16117 C4NL5R 10831793 Ki = 1500 nM T16117 CBYZ50 10840870 Ki = 4600 nM T16117 CJO21R 10845319 IC50 = 16000 nM T16117 CUID50 10849057 Ki = 29000 nM T16117 CC9A7Q 10852182 IC50 = 30000 nM T16117 CQ7A0W 10882498 IC50 = 13000 nM T16117 CB3CI1 10898715 IC50 = 1000 nM T16117 C93IGZ 10948273 IC50 = 34000 nM T16117 CDA0M4 10957874 IC50 = 6000 nM T16117 C8CLV2 10969874 IC50 = 42000 nM T16117 C1WY6T 11010340 IC50 = 60 nM T16117 CX5G2O 11013353 IC50 = 70000 nM T16117 CTL03M 11020380 IC50 = 1000 nM T16117 CK1JO5 11024952 IC50 = 44000 nM T16117 C0EK3A 11034111 IC50 = 40000 nM T16117 CM36UC 11058021 IC50 = 3300 nM T16117 C60TVY 11098403 IC50 = 50000 nM T16117 CJX3I6 11101028 IC50 = 11000 nM T16117 C3BVI2 11139807 IC50 = 3500 nM T16117 CH6Y1F 11149707 IC50 = 20000 nM T16117 CR0JK9 11159816 IC50 = 1300 nM T16117 C2X1GP 11161781 IC50 = 30000 nM T16117 C2BPQ8 11175135 IC50 = 141 nM T16117 C1CH0E 11194833 IC50 = 790 nM T16117 COC82L 11194834 IC50 = 350 nM T16117 C46FGL 11210360 IC50 = 123 nM T16117 COBY89 11229270 IC50 = 280 nM T16117 CAWM24 11240701 IC50 = 53 nM T16117 CQV6W7 11256080 IC50 = 112 nM T16117 CLN3E1 11267277 IC50 = 117 nM T16117 C6BM4C 11268382 IC50 = 96.3 nM T16117 CFN1Y0 11310025 IC50 = 6900 nM T16117 C5XS3F 11348978 IC50 = 161 nM T16117 CAH84T 11349572 IC50 = 39000 nM T16117 C6F7WD 11357119 IC50 > 100000 nM T16117 C8WF4O 11369870 IC50 = 96000 nM T16117 CTW93U 11390106 IC50 = 311000 nM T16117 CY03GF 11401263 IC50 = 280 nM T16117 CC98HE 11417668 IC50 = 330 nM T16117 CV97DZ 11426929 IC50 = 28000 nM T16117 C9SOQ7 11428573 IC50 = 121 nM T16117 CIK5B2 11438569 IC50 = 70.3 nM T16117 C0YOI9 11473924 IC50 = 390 nM T16117 C2AW4O 11480938 IC50 = 740 nM T16117 C10SLI 11480939 IC50 = 92 nM T16117 CHUP59 11481471 IC50 = 140000 nM T16117 CSBK19 11486109 IC50 = 203 nM T16117 CP84JR 11495366 EC50 > 100000 nM T16117 C1RU2I 11496223 EC50 = 310 nM T16117 CB43EZ 11502103 EC50 = 6000 nM T16117 CP7RX2 11523510 EC50 > 100000 nM T16117 C4JDI3 11524048 EC50 > 100000 nM T16117 CI8B3S 11531856 EC50 = 2700 nM T16117 C74RYA 11532340 EC50 > 100000 nM T16117 CO8SQ4 11532357 EC50 = 7600 nM T16117 C9F6KY 11538267 EC50 = 24000 nM T16117 CE1G4D 11539024 EC50 = 3900 nM T16117 C2KWX7 11546144 EC50 = 11000 nM T16117 CIEU85 11561546 EC50 = 690 nM T16117 CT1Z7W 11575808 EC50 > 100000 nM T16117 CWB4J7 11582528 EC50 = 9500 nM T16117 C09EFX 11589024 EC50 > 100000 nM T16117 CBR5I2 11590027 EC50 = 7200 nM T16117 C46KUP 11596038 EC50 > 100000 nM T16117 C2KVY7 11596934 EC50 = 6600 nM T16117 C0RTF7 11609610 EC50 > 100000 nM T16117 CDC1M2 11610728 EC50 > 100000 nM T16117 CK04AC 11624646 EC50 > 100000 nM T16117 CSI50Y 11625423 EC50 = 7200 nM T16117 C9E6TG 11631971 EC50 > 100000 nM T16117 C0MHE1 11633531 EC50 = 2100 nM T16117 CWG4J9 11639946 EC50 = 2300 nM T16117 CL7Q3I 11646432 EC50 = 17300 nM T16117 C4F0CK 11646596 EC50 > 100000 nM T16117 CA6D9Z 11654166 EC50 = 36000 nM T16117 C8UJ1K 11695590 EC50 > 100000 nM T16117 CM7YA3 11703771 EC50 > 100000 nM T16117 C8PZN0 11798374 Ki = 360 nM T16117 CDS16Y 11800991 Ki = 30600 nM T16117 C0TPY7 11827105 IC50 = 13000 nM T16117 CQ5RJ9 11957582 IC50 = 37000 nM T16117 CG63IC 12109769 IC50 > 100000 nM T16117 CBP7S2 12216463 Ki = 1000 nM T16117 CO7GP5 12297611 IC50 = 310000 nM T16117 C02XUH 12310464 Ki = 170000 nM T16117 CMHG98 12384935 Ki = 2000 nM T16117 CS5D0P 12404013 IC50 = 340 nM T16117 CLVQ03 12449028 IC50 > 100000 nM T16117 C2NX4W 12709336 IC50 > 50000 nM T16117 CNJ76X 12778905 IC50 = 20000 nM T16117 C4XK7S 12778908 IC50 = 400 nM T16117 CEJ53H 12778910 IC50 = 3500 nM T16117 CO7T1N 12969094 IC50 = 50000 nM T16117 CXA84F 13196077 IC50 > 50000 nM T16117 CZ2D9G 13268358 Ki = 8000 nM T16117 C9D4CW 13302397 IC50 = 10600 nM T16117 C9MC3D 13768254 IC50 = 3388.44 nM T16117 CI07KP 13768262 IC50 > 100000 nM T16117 C2L7PV 14833242 Ki = 8000 nM T16117 CZK9A7 15287360 IC50 = 610 nM T16117 C96DOX 15381020 IC50 = 13200 nM T16117 C7A2JC 15396734 Ki = 45000 nM T16117 CSJ32F 15453846 IC50 = 4500 nM T16117 C0O5LD 15453847 IC50 = 700 nM T16117 CAJF09 15512769 IC50 = 264 nM T16117 CHR3S4 15512781 IC50 = 137 nM T16117 C7RZ8B 15547276 Ki = 18000 nM T16117 CJ5H3U 15547277 Ki = 14000 nM T16117 CPF1W0 15871186 IC50 = 11000 nM T16117 COV8E5 15887952 IC50 = 5400 nM T16117 C2ZYA6 15951338 IC50 = 400 nM T16117 CL0SF3 15951408 IC50 = 350 nM T16117 C1Q8IV 15951410 IC50 = 540 nM T16117 CY9I5Z 16119079 IC50 > 200000 nM T16117 C6Z1DA 16739325 IC50 = 30 nM T16117 CD3CT0 17793169 IC50 = 11200 nM T16117 C9V0XQ 17897120 IC50 = 1310 nM T16117 C3X9JP 17958630 IC50 = 15720 nM T16117 CP2D3I 18356525 Ki = 40 nM T16117 C6RA2L 18414528 IC50 = 350 nM T16117 CKMV50 18428554 IC50 = 1600 nM T16117 CMSA79 18687946 Ki = 1000 nM T16117 C05KOC 18721714 IC50 > 50000 nM T16117 C98OVY 18721715 IC50 = 25890 nM T16117 CY28GR 18721729 IC50 > 50000 nM T16117 CY7EO4 18800758 IC50 = 12100 nM T16117 CW0IX3 18983434 IC50 = 53000 nM T16117 CFB10N 20102781 IC50 = 11500 nM T16117 CQZ84B 21192814 IC50 = 1000 nM T16117 CN5A8J 21834414 IC50 = 2400 nM T16117 CW2VK6 21878467 IC50 = 200 nM T16117 CH70CD 22133392 IC50 > 100000 nM T16117 CH3SV2 23218983 Ki = 75000 nM T16117 CZ3X6F 24745386 Ki = 13000 nM T16117 CBNT78 24745536 Ki = 10000 nM T16117 CN1D9J 24758920 IC50 = 130 nM T16117 CPH67W 24764596 Ki = 5.3 nM T16117 C02RPF 24782142 EC50 = 690 nM T16117 C2UR8E 24782146 EC50 > 10000 nM T16117 C74IOP 24782646 EC50 > 10000 nM T16117 C40NIF 24782649 EC50 > 10000 nM T16117 CD2T4M 24782902 EC50 > 10000 nM T16117 CFG23E 24782903 EC50 = 1500 nM T16117 CM50WK 24785172 EC50 > 10000 nM T16117 C6U0PV 24785174 EC50 = 690 nM T16117 CD7K3S 24785426 EC50 > 10000 nM T16117 CT2UV6 24785697 EC50 = 650 nM T16117 C3MWU8 24785698 EC50 = 770 nM T16117 CWK68M 24785700 EC50 = 320 nM T16117 C4TC8F 24785702 EC50 = 5000 nM T16117 CO65CH 24785966 EC50 > 100000 nM T16117 CTLA48 24785968 EC50 = 990 nM T16117 C5VBE0 24787679 IC50 = 7900000 nM T16117 CPN5Z3 24798097 Ki = 0.085 nM T16117 C86KAI 24798098 Ki = 52 nM T16117 C7IXF0 24850786 Ki = 0.388 nM T16117 CFJX70 24850913 Ki = 9.4 nM T16117 CPQ15V 24894148 IC50 = 3100 nM T16117 CYU1V8 24894149 IC50 = 7800 nM T16117 CNX5Q3 24894150 IC50 = 100000 nM T16117 C3QK6V 24894151 IC50 = 63000 nM T16117 C6J0NK 24894153 IC50 = 80 nM T16117 C7Q3YX 24894154 IC50 = 50 nM T16117 CV7M1Y 24936091 IC50 = 5300 nM T16117 C7DM6Y 25021186 Ki = 0.25 nM T16117 CR3I9Y 25050394 EC50 = 3200 nM T16117 C39DOQ 25050395 EC50 > 10000 nM T16117 CW0Q3F 25210996 EC50 = 520 nM T16117 C9T1XJ 25211376 EC50 = 1300 nM T16117 CD09PR 25211378 EC50 = 1600 nM T16117 CD0F1I 25211400 IC50 = 330 nM T16117 C5K3ZC 25211401 IC50 = 120 nM T16117 C9O3QC 25211403 IC50 = 60 nM T16117 CSG69X 25211404 IC50 = 64 nM T16117 CF79GW 25211493 EC50 = 760 nM T16117 CE9DK7 25211494 EC50 = 1000 nM T16117 C0DOS1 25211596 EC50 = 1300 nM T16117 CT3ID6 25211597 EC50 = 2000 nM T16117 C2UQJ6 25211598 EC50 = 300 nM T16117 C43HVC 25211599 EC50 = 1000 nM T16117 CDV7E8 25211804 EC50 = 6800 nM T16117 CKI86X 25211805 EC50 = 4600 nM T16117 CHW2X0 25211910 EC50 = 300 nM T16117 CW0Q7Y 25212125 IC50 = 100 nM T16117 C4EF2A 25212418 IC50 = 46 nM T16117 CNV40T 42618036 EC50 > 10000 nM T16117 CH7AS5 42618037 EC50 > 10000 nM T16117 C97FDE 42618038 EC50 > 10000 nM T16117 C3MJQ4 42618039 EC50 > 10000 nM T16117 C1YO7H 42618040 EC50 = 2300 nM T16117 C0B6JO 42618041 EC50 > 10000 nM T16117 C3G6HZ 42618043 EC50 = 2700 nM T16117 C3C4FA 42618044 EC50 > 10000 nM T16117 C2SK5R 42618045 EC50 > 10000 nM T16117 C1V0KI 42618047 EC50 = 7900 nM T16117 CXE5C2 42618048 EC50 = 2100 nM T16117 C3S4NL 42618049 EC50 = 2200 nM T16117 CN6WQ5 42618050 EC50 = 4100 nM T16117 C5F6PW 42618052 EC50 = 500 nM T16117 CMQI75 42618053 EC50 = 10300 nM T16117 CN34WV 42618054 EC50 = 2900 nM T16117 CH81PY 42618060 EC50 > 10000 nM T16117 C4QS7B 42618062 EC50 > 10000 nM T16117 CAZ25X 42618063 EC50 = 3400 nM T16117 CX5NI3 42618064 EC50 > 10000 nM T16117 C54TBN 42618065 EC50 > 10000 nM T16117 C0I4MK 42618066 EC50 = 120 nM T16117 CGU3N8 42618068 EC50 = 70 nM T16117 C5UN1C 42618069 EC50 = 97 nM T16117 C8JFX2 42618070 EC50 > 10000 nM T16117 CRQ96D 42634153 IC50 = 1420 nM T16117 CGY1S0 44291051 Ki = 330 nM T16117 C9C5TH 44294245 Ki = 8400 nM T16117 CKT5C3 44294421 Ki = 29000 nM T16117 CYI6D2 44302109 IC50 = 160 nM T16117 CE9LX0 44302114 IC50 = 140 nM T16117 CR5C8Z 44302148 IC50 = 170 nM T16117 C1T7UQ 44302150 IC50 = 170 nM T16117 C2YDZ6 44319656 IC50 = 110 nM T16117 CQYW59 44319709 IC50 = 730 nM T16117 CO1Z2F 44319710 IC50 = 680 nM T16117 C54VXO 44319711 IC50 = 240 nM T16117 CUY6V5 44319750 IC50 > 100000 nM T16117 CMU93E 44319752 IC50 = 100000 nM T16117 C5M9IL 44319753 IC50 = 6800 nM T16117 CA81IQ 44319778 IC50 = 310 nM T16117 CD1QB5 44319779 IC50 = 130 nM T16117 CR3HT4 44319780 IC50 = 500 nM T16117 C59RGW 44319825 IC50 = 130 nM T16117 C76IJF 44319826 IC50 = 190 nM T16117 CY8K0G 44319828 IC50 = 640 nM T16117 CQ5A4R 44320031 IC50 = 640 nM T16117 C0PQ4L 44320069 IC50 = 4100 nM T16117 CL42AK 44320084 IC50 = 1600 nM T16117 C9M6VH 44320114 IC50 = 3300 nM T16117 CV4XW8 44320115 IC50 = 2100 nM T16117 CHT83A 44320347 IC50 = 212 nM T16117 C80ORG 44322605 IC50 = 108000 nM T16117 C1O4FX 44323742 Ki = 450 nM T16117 C1UJH7 44326624 Ki = 12000 nM T16117 C45LQR 44326626 Ki = 60000 nM T16117 CMH1Y0 44326628 Ki = 50000 nM T16117 CD43JV 44326650 Ki = 10000 nM T16117 CL4AK3 44326665 Ki = 6000 nM T16117 CPDW12 44326817 Ki = 45000 nM T16117 C1VZD7 44326869 Ki = 14000 nM T16117 C6N4GL 44326871 Ki = 3000 nM T16117 C8WN9I 44327898 Ki = 9300 nM T16117 CCM47P 44328869 Ki = 56 nM T16117 CZ2BS4 44328871 Ki = 170 nM T16117 C7FG5O 44328879 Ki = 14000 nM T16117 C4N5IJ 44328899 Ki = 29000 nM T16117 C34CQV 44328929 Ki = 39000 nM T16117 C0BDZ8 44328932 Ki = 5600 nM T16117 CSG52F 44328934 Ki > 50000 nM T16117 CDF12B 44328946 Ki = 7200 nM T16117 CVO68P 44328955 Ki = 13000 nM T16117 CTAF63 44328957 Ki = 33000 nM T16117 C0W1JK 44328968 Ki = 600 nM T16117 C7GS5O 44328973 Ki = 2100 nM T16117 C14UCS 44328998 Ki > 50000 nM T16117 CEP9D7 44329003 Ki = 1500 nM T16117 CZQ78B 44329038 Ki = 360 nM T16117 CG6F2P 44329061 Ki = 14000 nM T16117 C8UEJ6 44329070 Ki = 1100 nM T16117 C39GJB 44329072 Ki = 7500 nM T16117 CPOB75 44329074 Ki > 50000 nM T16117 C3OUZ7 44329119 Ki = 570 nM T16117 CMW2I5 44329128 Ki = 4600 nM T16117 CNZ5T9 44329167 Ki = 46000 nM T16117 CP4ZU0 44329169 Ki > 50000 nM T16117 CW1VT4 44329187 Ki > 50000 nM T16117 C7PG5J 44329191 Ki > 50000 nM T16117 C1TKS5 44329193 Ki = 11000 nM T16117 C86AGM 44329195 Ki = 2800 nM T16117 C25XJI 44329227 Ki = 370 nM T16117 CV67AL 44329240 Ki = 4600 nM T16117 CEBZ52 44329255 Ki = 42 nM T16117 CYX4T3 44329820 IC50 = 50000 nM T16117 C1FHY4 44329948 IC50 = 4400 nM T16117 C5W4FL 44329963 IC50 = 4400 nM T16117 CBQ1O0 44329995 IC50 = 68000 nM T16117 C01SEL 44331035 IC50 = 48000 nM T16117 CS1F8K 44331045 IC50 = 192000 nM T16117 CHJG24 44331075 IC50 = 180000 nM T16117 CG4IJ0 44331086 IC50 = 94000 nM T16117 C9JNB4 44331280 IC50 = 300000 nM T16117 CE40MJ 44331339 IC50 = 8000 nM T16117 CB70RG 44331486 Ki = 580 nM T16117 C94MNS 44336772 Ki = 1700 nM T16117 CQ81IY 44336958 Ki = 770 nM T16117 C9GC1B 44337005 Ki = 1100 nM T16117 CK7SD9 44337020 Ki = 320 nM T16117 C8F5EQ 44341087 IC50 = 49000 nM T16117 CQ0CU9 44341212 IC50 = 240 nM T16117 CU62NQ 44341315 IC50 = 20000 nM T16117 CWQ18O 44341316 IC50 = 8900 nM T16117 C2YC1E 44347417 IC50 = 2530 nM T16117 C86PTS 44347432 IC50 = 850 nM T16117 C3OV4R 44368785 Ki = 890 nM T16117 CQ6DG0 44370661 IC50 > 100000 nM T16117 C0FRX8 44370662 IC50 > 100000 nM T16117 C46TVU 44370689 IC50 > 100000 nM T16117 CYI91R 44370690 IC50 > 100000 nM T16117 C9GZB5 44370704 IC50 > 100000 nM T16117 CKQ20Y 44370705 IC50 = 6000 nM T16117 CS4M3D 44370729 IC50 = 630000 nM T16117 CI7K3E 44370730 IC50 = 53000 nM T16117 C6VS9A 44370736 IC50 = 68000 nM T16117 C12SON 44370747 IC50 = 11600 nM T16117 CF5W2Z 44377082 IC50 = 590 nM T16117 CW0F6J 44377099 IC50 = 310 nM T16117 C7K8XO 44377152 IC50 = 660 nM T16117 C6C2YV 44377153 IC50 = 290 nM T16117 C2NZ1X 44393481 IC50 > 50000 nM T16117 CDSJ39 44393485 IC50 = 14000 nM T16117 C10WEK 44393495 IC50 > 50000 nM T16117 C3GDF7 44393630 IC50 = 75 nM T16117 C9M5SP 44393639 IC50 = 200 nM T16117 C6CDT1 44393666 IC50 = 235 nM T16117 CTD27K 44393700 IC50 = 75 nM T16117 CJ02FD 44393705 IC50 = 112 nM T16117 C93KUZ 44393711 IC50 = 810 nM T16117 C85GFC 44396192 IC50 > 50000 nM T16117 C4XL3B 44399796 IC50 = 1300 nM T16117 C53KME 44399834 IC50 = 610 nM T16117 CU98HN 44399945 IC50 = 190 nM T16117 CYW0O2 44400067 IC50 = 240 nM T16117 CU6M4D 44402389 IC50 = 38000 nM T16117 C94GAW 44402453 IC50 > 1000000 nM T16117 CDIR71 44402600 IC50 = 3500 nM T16117 CQTC93 44402628 IC50 = 500000 nM T16117 CL5I8G 44430315 IC50 = 42 nM T16117 CEH14S 44430628 IC50 = 1100 nM T16117 C0WX4U 44430629 IC50 = 1300 nM T16117 CUO30Z 44430631 IC50 = 400 nM T16117 C90QJT 44430632 IC50 = 800 nM T16117 CLZ51V 44430633 IC50 = 200 nM T16117 CWT98D 44430634 IC50 = 300 nM T16117 C62UWN 44430635 IC50 = 4400 nM T16117 CI8WV0 44430636 IC50 = 2000 nM T16117 CG13ZP 44430637 IC50 = 100 nM T16117 C43QST 44430638 IC50 = 200 nM T16117 C8PTS2 44430640 IC50 = 300 nM T16117 C58QXR 44430641 IC50 = 5100 nM T16117 CRF8W4 44455594 IC50 = 4900 nM T16117 C2Z5TD 44455595 IC50 = 6500 nM T16117 CUK8X2 44455597 IC50 = 1200 nM T16117 C4PE7R 44455626 IC50 = 1200 nM T16117 C1E3AV 44455627 IC50 = 1200 nM T16117 C05FUP 44455628 IC50 = 2500 nM T16117 C4UZH5 44455631 IC50 = 190 nM T16117 CSOK53 44455662 IC50 = 1900 nM T16117 C34XKU 44455663 IC50 = 748 nM T16117 C50IWU 44455685 IC50 = 190 nM T16117 C9E7NX 44455718 IC50 = 150 nM T16117 CH9W2F 44455719 IC50 = 360 nM T16117 CG6I8D 44455720 IC50 = 140 nM T16117 CV8JE9 44455746 IC50 = 600 nM T16117 CEGL71 44455747 IC50 = 530 nM T16117 C8DQV4 44455748 IC50 = 1800 nM T16117 CHAZ31 44455749 IC50 = 420 nM T16117 CPDZ45 44455769 IC50 = 370 nM T16117 C02SZW 44455770 IC50 = 810 nM T16117 CQ2VA3 44455771 IC50 = 350 nM T16117 C6CYN7 44455794 IC50 = 590 nM T16117 CVMY02 44455795 IC50 = 530 nM T16117 CN3D9Q 44455797 IC50 = 780 nM T16117 CSIX74 44455821 IC50 = 540 nM T16117 C03BYA 44565909 EC50 = 360 nM T16117 C8DUG3 44566070 EC50 = 290 nM T16117 C32ARX 44586238 Ki = 94000 nM T16117 C24VGQ 44586264 Ki = 35000 nM T16117 C0BQC4 44586265 Ki = 60000 nM T16117 CG09ZB 44586266 Ki = 2000 nM T16117 C2W6GB 44586267 Ki = 65000 nM T16117 C8RY0A 44586268 Ki = 2000 nM T16117 C86RGB 44586304 Ki = 150000 nM T16117 C8HB7X 44586305 Ki = 80000 nM T16117 C34DOU 44586306 Ki = 100000 nM T16117 C59ENX 44586307 Ki = 70000 nM T16117 CL63WE 44586561 Ki = 4800 nM T16117 CIFH20 44592963 IC50 = 15300 nM T16117 CAY89U 44592964 IC50 = 4000 nM T16117 CW2VG0 44592965 IC50 = 12200 nM T16117 CH6R7D 44592966 IC50 = 700 nM T16117 C2AMT5 44592991 IC50 = 4200 nM T16117 CHP0I9 44592992 IC50 = 700 nM T16117 C9ASJ2 44592993 IC50 = 6600 nM T16117 CPT86N 44592994 IC50 = 3000 nM T16117 CGNO91 46225774 Ki = 50 nM T16117 CZ5E0N 46847260 IC50 = 5000 nM T16117 CN51IS 46880969 IC50 = 10000 nM T16117 C8J6ZT 46880970 IC50 = 19000 nM T16117 CK03TN 46907789 Ki = 290 nM T16117 CGU7K3 46907790 Ki = 1800 nM T16117 CB1Y8N 49796134 IC50 > 1850000 nM T16117 CN8T5X 49796514 IC50 = 27000 nM T16117 CE24XP 49831165 Ki = 490 nM T16117 CM2D5Z 49836940 EC50 = 4300 nM T16117 CZ51GS 49836941 EC50 > 10000 nM T16117 CM2JB5 49836942 EC50 = 2900 nM T16117 C6ZA7M 49836943 EC50 = 650 nM T16117 C1IHW8 49836944 EC50 = 1400 nM T16117 CM10KE 49837060 EC50 = 950 nM T16117 C3J2SH 49837061 EC50 = 650 nM T16117 CP92KI 49837062 EC50 = 24000 nM T16117 C2ZD0V 49837063 EC50 = 730 nM T16117 C1SB6T 49837065 EC50 = 610 nM T16117 CK38CR 49837066 EC50 = 1100 nM T16117 CD8GN9 49837170 EC50 = 3000 nM T16117 CVC18N 49861985 Ki = 130 nM T16117 CZJ85F 49864405 IC50 = 1000 nM T16117 C1MYW7 53233132 IC50 = 14000 nM T16117 CZWO31 53387025 IC50 = 98 nM T16117 C6AYE3 53392451 IC50 = 130 nM T16117 CQ8W0K 54580275 IC50 = 1700 nM T16117 C6TN1Y 54583301 IC50 > 100000 nM T16117 C6QK1A 56593711 IC50 = 200 nM T16117 CXSQ19 56593712 IC50 = 800 nM T16117 CY70WM 56593713 IC50 = 120 nM T16117 C48VIC 56593714 IC50 = 1500 nM T16117 C4U6BD 56593857 IC50 = 450 nM T16117 CC86JF 56659406 IC50 = 446.68 nM T16117 CSBN93 56659435 IC50 = 6606.93 nM T16117 C6P5YB 56666339 IC50 > 100000 nM T16117 CDF86T 56669739 IC50 = 1905.46 nM T16117 CRZ08C 56673237 IC50 = 58884.37 nM T16117 C8TA3D 56679900 IC50 > 100000 nM T16117 C73MZW 56924689 IC50 = 370 nM T16117 C83REA 56949933 IC50 = 4070 nM T16117 C2DJ7A 56949934 IC50 = 3260 nM T16117 C3B4DI 56949935 IC50 = 2070 nM T16117 C5DK8C 56950062 IC50 = 110 nM T16117 C13TGD 56950064 IC50 = 70 nM T16117 CF2VW1 56950067 IC50 = 180 nM T16117 CHO6F5 56950186 IC50 = 540 nM T16117 CHQ5S6 56950187 IC50 = 18800 nM T16117 CRG42P 56950331 IC50 = 5750 nM T16117 C6BZ7V 56951568 IC50 = 12 nM T16117 C0UW5Z 57341142 IC50 = 97 nM T16117 CS2FH5 57341143 IC50 = 133 nM T16117 C2AUM9 57341144 IC50 = 176 nM T16117 CX1FQ0 57341332 IC50 = 235 nM T16117 CN3Y9D 57341333 IC50 = 139 nM T16117 C3H1GV 57341334 IC50 = 267 nM T16117 C0Z3JI 57341335 IC50 = 115 nM T16117 C83DHY 57341336 IC50 = 248 nM T16117 CDU9W0 57341337 IC50 = 169 nM T16117 CBO89M 57384807 IC50 = 840 nM T16117 C2BAZ9 57385041 IC50 = 1730 nM T16117 C2TAS4 57385549 IC50 = 300 nM T16117 CX2TG9 57385550 IC50 = 490 nM T16117 CVM67R 57385790 IC50 = 200 nM T16117 COQ83X 57391112 EC50 = 18000 nM T16117 C19RIY 57391700 IC50 = 370 nM T16117 CB1NH9 57392807 EC50 > 100000 nM T16117 C6FD9C 57393301 IC50 = 213 nM T16117 C7TM3R 57393317 IC50 = 130 nM T16117 C6RKY7 57393439 IC50 = 1600 nM T16117 C5QMZ6 57393919 IC50 = 950 nM T16117 C21UDR 57394528 EC50 > 100000 nM T16117 CVC7Z2 57394614 EC50 = 11000 nM T16117 CPQ0S7 57394615 EC50 = 7900 nM T16117 C9J6IM 57395031 IC50 = 160 nM T16117 CP4TV8 57395168 IC50 = 170 nM T16117 COKU75 57396367 EC50 > 100000 nM T16117 CV7HI9 57396371 EC50 = 480 nM T16117 CL0P6T 57396785 IC50 = 440 nM T16117 C2QS6D 57396941 IC50 = 69 nM T16117 C4BO9G 57398563 IC50 = 62 nM T16117 C1DCN7 57401588 EC50 = 47000 nM T16117 CQ5HU7 57401590 EC50 > 100000 nM T16117 CI2DY9 57403339 EC50 = 6800 nM T16117 CD9P4Z 57403764 IC50 = 500 nM T16117 C2ONF1 57403909 IC50 = 240 nM T16117 CYQ70T 57403910 IC50 = 360 nM T16117 CM6C1O 57403911 IC50 = 150 nM T16117 CSWV56 57474449 IC50 = 1290 nM T16117 C0L5HT 62706594 IC50 = 440 nM T16117 CJHB32 62706595 IC50 = 740 nM T16117 C9EIX4 62706596 IC50 = 1770 nM T16117 C04WBM 62706597 IC50 = 12800 nM T16117 CS9KV1 62706598 IC50 = 5050 nM T16117 CX72ZW 62706764 IC50 = 2760 nM T16117 C24YCI 62706765 IC50 = 14400 nM T16117 CEL48Q 62706766 IC50 > 100000 nM T16117 C7XEA4 62706767 IC50 = 35700 nM T16117 CC5B6H 62706768 IC50 = 37200 nM T16117 CO7AH9 66912415 IC50 = 450 nM T16117 CA7DI2 66912425 IC50 = 150 nM T16117 C2PK8Q 66912454 IC50 = 1400 nM T16117 C37DOA 66912484 IC50 = 1000 nM T16117 C78AWC 66912498 IC50 = 2730 nM T16117 C8Y7AV 66912516 IC50 = 1780 nM T16117 CPB9C5 66912809 IC50 = 2400 nM T16117 CF0J3M 67340183 IC50 = 660 nM T16117 C5HSI6 67492912 IC50 = 110 nM T16117 C9FMX2 67493358 IC50 = 440 nM T16117 C7ME1A 70682896 Ki = 2000 nM T16117 C3UO2F 70686000 IC50 = 1370 nM T16117 CWO02R 70688127 IC50 = 730 nM T16117 C16YWC 71454528 Ki = 1250 nM T16117 C0M6DH 71484435 IC50 = 100 nM T16117 CIE6A1 71486265 IC50 = 40 nM T16117 C2Y1CX 71486266 IC50 = 120 nM T16117 CO8D6C 71486267 IC50 = 620 nM T16117 C19AXY 71486268 IC50 = 350 nM T16117 CK0SO4 71486403 IC50 = 80 nM T16117 C2C0RP 71486404 IC50 = 430 nM T16117 CS0X2Q 71486405 IC50 = 160 nM T16117 C7DH8X 71486406 IC50 = 200 nM T16117 C9VIN3 71486407 IC50 = 690 nM T16117 CRZ73J 71486408 IC50 = 330 nM T16117 CW9V2Q 71718237 IC50 = 35 nM T16117 CM1DB0 71719440 IC50 = 140 nM T16117 CX5O2N 71724308 IC50 = 880000 nM T16117 CQ97HX 71724310 IC50 = 530000 nM T16117 C4Z9PQ 71724455 IC50 = 400000 nM T16117 CC6Q5R 72771081 Ki = 440 nM T16117 C0TSY5 72771082 Ki = 318 nM T16117 CXZ71D 76033629 IC50 = 1050 nM T16117 C1B5YU 78426481 Ki = 318 nM T16117 CX41AE 78426482 Ki = 440 nM T16117 CWD54N 86767080 Ki = 90 nM T16117 C26ADC 90662876 IC50 = 430 nM T16117 C3QU2O 90662877 IC50 = 320 nM T16117 CYUW16 90664333 IC50 = 760 nM T16117 CRK93Y 90664334 IC50 = 360 nM T16117 CAUK54 90664335 IC50 = 170 nM T16117 CR35FV 90664340 IC50 = 160 nM T16117 CZ8H2M 90664341 IC50 = 1220 nM T16117 C5UNM2 90664342 IC50 = 270 nM T16117 CE5H8T 90664346 IC50 = 2380 nM T16117 CVY3L6 90664347 IC50 = 330 nM T16117 CPNS27 90664349 IC50 = 113000 nM T16117 C5RHW1 90664461 IC50 = 360 nM T16117 CRX47I 90664467 IC50 = 18000 nM T16117 CNLO43 90664468 IC50 = 14000 nM T16117 C2G0XJ 90664469 IC50 = 2250 nM T16117 CU7Q9V 90664588 IC50 = 1220 nM T16117 C9TLX0 90664602 IC50 = 70 nM T16117 C7JIW4 90664606 IC50 = 360 nM T16117 CP1JM7 90664607 IC50 = 10400 nM T16117 CN7P3V 90664608 IC50 = 160 nM T16117 C8LFX7 90664695 IC50 = 200 nM T16117 CU29TX 90664696 IC50 = 520 nM T16117 C7FQ5W 90664698 IC50 = 700 nM T16117 C8X1LA 90664704 IC50 = 250 nM T16117 C1PHN4 90664711 IC50 = 1200 nM T16117 C6EGO9 90664714 IC50 = 260 nM T16117 CS65XI 90664715 IC50 = 170 nM T16117 CJ61NW 90664716 IC50 = 20 nM T16117 CQT69X 90664721 IC50 = 430 nM T16117 CVXO58 90664722 IC50 = 260 nM T16117 CUNK69 90664723 IC50 = 86 nM T16117 CE7H6D 90664727 IC50 = 2240 nM T16117 C9Y2FD 90664833 IC50 = 220 nM T16117 CE3RV1 90664839 IC50 = 2210 nM T16117 CGK56Q 90664840 IC50 = 780 nM T16117 C0JM7D 90664841 IC50 = 1140 nM T16117 CL0TG4 90664842 IC50 = 93 nM T16117 CN3A1P 90664848 IC50 = 550 nM T16117 C7H8FN 90664849 IC50 = 1960 nM T16117 CA81EW 90664850 IC50 = 2960 nM T16117 C7HGP1 90664855 IC50 = 80 nM T16117 CYI01T 90664884 Ki = 493 nM T16117 C8F7HI 90664950 IC50 = 260 nM T16117 CHA2T6 90664963 IC50 = 90 nM T16117 CJ01LW 90664969 IC50 = 580 nM T16117 C8PCH5 90664970 IC50 = 3360 nM T16117 CYT2F5 90664975 IC50 = 4830 nM T16117 CUD3G0 90665016 Ki = 440 nM T16117 C5FZK7 90665071 IC50 = 870 nM T16117 CF14BZ 90665089 IC50 = 410 nM T16117 CI4H7Y 90665090 IC50 = 490 nM T16117 C7PHT4 90665099 IC50 = 1020 nM T16117 C0LM7T 90665100 IC50 = 1860 nM T16117 CY4F6W 90665101 IC50 = 100 nM T16117 C57NEK 90665196 IC50 = 120 nM T16117 C3E6MO 90665203 IC50 = 470 nM T16117 C79CZW 90665204 IC50 = 60 nM T16117 C2WUY8 90665205 IC50 = 950 nM T16117 CK62BX 90665207 IC50 = 820 nM T16117 C02PLA 90665208 IC50 = 540 nM T16117 CB63ER 90665216 IC50 = 190 nM T16117 CS8NH6 91808024 Ki = 98 nM T16117 C4IG3X 91808025 Ki = 64 nM T16117 C8HLF9 91808026 Ki = 55 nM T16117 CR93ZO 91808031 Ki = 59 nM T16117 CU43ZF 91819607 Ki = 189 nM T16117 C1DF0K 91819608 Ki = 105 nM T16117 CQ35RI 91971384 Ki = 911 nM T16117 CB0A4F 91971388 Ki = 295 nM T16117 CL8F9S 118266141 Ki = 768 nM T16117 CK1MG8 118730368 Ki = 758 nM T16117 CTE58Z 118730369 Ki = 193 nM T16117 CQ1S4F 118730370 Ki = 125 nM T16117 C9N1ZG 118730371 Ki = 359 nM T16117 CQT3Y0 118730372 Ki = 358 nM T16117 C1PR2Q 118730373 Ki = 125 nM T16117 CB36KU 118730374 Ki = 138 nM T16117 C52QGJ 118730382 Ki = 303 nM T16117 C4EI0W 118730384 Ki = 137 nM T16117 C7O8RE 118730386 Ki = 873 nM T16117 C6JP8E 119057273 Ki = 84 nM T16117 C1MFO5 119057274 Ki = 89 nM T16117 COLQ09 119081686 Ki = 862 nM T16117 CL3DK1 119081688 Ki = 13 nM T16117 CUD7Q0 119081689 Ki = 37 nM T16117 C0YD5S 121250392 Ki = 50 nM T16117 CL98KI 121250394 Ki = 32 nM T16117 CZM87C 121250396 Ki = 20 nM T16117 CEA5V4 121250401 Ki = 52 nM T16117 C6EH9G 121250403 Ki = 21 nM T16117 CTQ9U6 121250406 Ki = 30 nM T16117 C2HZ3T 121262516 Ki = 764 nM T16117 CZ63FM 121262521 Ki = 76 nM T16117 CL82JK 121262526 Ki = 164 nM T16117 CG8L4W 121312090 Ki = 109 nM T16117 CYN8X3 121312091 Ki = 56 nM T16117 CY5LD2 121596956 Ki = 1020 nM T16117 CRTW41 121596957 Ki = 108 nM T16117 CS6C3O 122180513 Ki = 111 nM T16117 CH7Q5A 124136836 Ki = 33 nM T16117 CG0EN1 124136841 Ki = 74 nM T16117 CF70JE 124136845 Ki = 61 nM T16117 CRPM16 124136846 Ki = 51 nM T16117 C7JLU1 124136856 Ki = 78 nM T16117 CD24UM 124136858 Ki = 31 nM T16117 CD54ZK 124136869 Ki = 136 nM T16117 CLZ38Y 124136872 Ki = 65 nM T16117 CG0HT3 124136874 Ki = 52 nM T16117 CP95UD 124136876 Ki = 36 nM T16117 CHOG43 124136880 Ki = 54 nM T16117 C8E1MD 124136896 Ki = 125 nM T16117 C7ONE0 124136898 Ki = 56 nM T16117 CT2PQ8 124136901 Ki = 46 nM T16117 CM49SP 124145844 Ki = 274 nM T16117 CH5GX6 124145845 Ki = 73 nM T16117 C1C0KT 124145846 Ki = 4300 nM T16117 CCG20T 124145847 Ki = 1100 nM T16117 C3MKV2 124145848 Ki = 2050 nM T16117 C0S7KT 124145849 Ki = 130 nM T16117 C27WCY 127034886 Ki = 1860 nM T16117 CNF3Z6 127034888 Ki = 855 nM T16117 C4PJN1 127034889 Ki = 911 nM T16117 CZ07EI 127034910 Ki = 1080 nM T16117 CR61YN 127034912 Ki = 295 nM T16117 CO3PW5 127034913 Ki = 507 nM T16117 CU61CX 127035691 Ki = 657 nM T16117 C7C9DU 127046260 IC50 = 180000 nM T16117 C6HI1S 127047637 IC50 > 1000000 nM T16117 CQI26T 127047755 IC50 > 1000000 nM T16117 C9QJ2I 127047967 IC50 = 800000 nM T16117 CIO56U 127047968 IC50 = 860000 nM T16117 CCGY27 127048125 IC50 > 1000000 nM T16117 CS9E0R 127050046 Ki = 425 nM T16117 C1UK4S 129168339 Ki = 2170 nM T16117 CL2YX7 130449136 Ki = 65 nM T16117 C1UTC8 130449148 Ki = 55 nM T16117 CTL8B5 130449158 Ki = 30 nM T16117 CV41FA 130449315 Ki = 43 nM T16117 C7J9BX 134686794 Ki = 516 nM T16117 C6OGU3 134686796 Ki = 82 nM T16117 C0A9BD 134686797 Ki = 100 nM T16117 CGX96C 134686798 Ki = 83 nM T16117 CXL4V8 135409388 IC50 = 7300 nM T16117 C76NBO 135409922 IC50 = 20000 nM T16117 CHKO08 135420615 IC50 = 145000 nM T16117 C83ZLX 135449023 IC50 = 22350 nM T16117 C7O9XT 135458572 IC50 > 100000 nM T16117 C5VD4I 135464339 IC50 = 60000 nM T16117 C47IWU 135470444 IC50 = 28000 nM T16117 C72AKJ 135480132 IC50 = 44000 nM T16117 C1S4KM 135490493 IC50 = 42000 nM T16117 CM8XF5 135502005 IC50 = 26000 nM T16117 COH6F0 135511896 IC50 = 50000 nM T16117 C2FJ6G 135519036 IC50 = 650000 nM T16117 CHN4Y9 135529990 IC50 = 190000 nM T16117 C5H2QR 135674618 IC50 > 500000 nM T16117 C8MN2E 135973134 IC50 = 8000 nM T16117 CT9K3I 136026480 IC50 > 100000 nM T16117 CGKE32 136035291 IC50 = 29000 nM T16117 CJ9M6N 136035292 IC50 = 88000 nM T16117 C7WPI2 136035293 IC50 = 38000 nM T16117 CWJ17V 136035300 IC50 = 81000 nM T16117 CMCS36 136035301 IC50 = 16000 nM T16117 CPC52T 136035302 IC50 = 90000 nM T16117 C46TCX 136035303 IC50 = 125000 nM T16117 CIJ10U 136035304 IC50 = 40000 nM T16117 C7ZU2K 136035305 IC50 = 130000 nM T16117 CK9LR3 136035306 IC50 = 8000 nM T16117 C59LGM 136035307 IC50 = 32000 nM T16117 CN7KB4 136035308 IC50 = 63000 nM T16117 C3GC5N 136035309 IC50 = 172000 nM T16117 CWPC96 136035310 IC50 = 25000 nM T16117 C0DA9Q 136035311 IC50 = 42000 nM T16117 CKO72Q 136035312 IC50 = 46000 nM T16117 C31TUI 136035313 IC50 = 21000 nM T16117 CTJ0I9 136035316 IC50 = 30000 nM T16117 COA8D6 136109078 IC50 = 116900 nM T16117 CHC62Q 136109080 IC50 = 85100 nM T16117 CB4UO8 136109082 IC50 = 33460 nM T16117 CG7JZ4 137530108 Ki = 58 nM T16117 COR09H 137530109 Ki = 124 nM T16117 CG9TL7 137530110 Ki = 68 nM T16117 CFZ74Y 137530111 Ki = 52 nM T16117 CD43TC 137530112 Ki = 59 nM T16117 CM6C7Y 137530113 Ki = 204 nM T16117 CL41DA 137530114 Ki = 29 nM T16117 C4AJP1 137530115 Ki = 36 nM T16117 CULW10 137530116 Ki = 157 nM T16117 CW7V4O 137530117 Ki = 58 nM T16117 C9USH3 137530118 Ki = 46 nM T16117 CDKB20 137530119 Ki = 43 nM T16117 CSR3F0 137530120 Ki = 37 nM T16117 CA39SN 137530121 Ki = 21 nM T16117 CH26CO 137530122 Ki = 89 nM T16117 CCH10Y 137530123 Ki = 84 nM T16117 CP3DL2 137530124 Ki = 129 nM T16117 CDLF21 137530125 Ki = 87 nM T16117 CH1S5L 137530126 Ki = 23 nM T16117 CDOS52 137633546 Ki = 598 nM T16117 C95OYQ 137637529 Ki = 362 nM T16117 CAN9G4 146025971 Ki = 111 nM T16117 CMTI65 146025972 Ki = 58 nM T16117 CN6H0M 146025973 Ki = 66 nM T16117 CQ9P2B 146025974 Ki = 96 nM T16117 CN8JM9 146025975 Ki = 46 nM T16117 CYOA91 146025976 Ki = 76 nM T16117 CS0BW8 146025977 Ki = 45 nM T16117 CY37WD 146025978 Ki = 31 nM T16117 C4S1ZP 146025979 Ki = 63 nM T16117 C8RWQ4 146025980 Ki = 46 nM T16117 C9R5SN 146025981 Ki = 114 nM T16117 CCP8X4 155513324 Ki = 151 nM T16117 COL57U 155518596 Ki = 149 nM T16117 CG35TK 155527043 Ki = 122 nM T16117 CZEY25 155533249 Ki = 106 nM T16117 CF85SO 155534420 Ki = 72 nM T16117 C7ZTA4 155540835 Ki = 60 nM T16117 COAM39 155543079 Ki = 88 nM T16117 CE8YT1 155563274 Ki = 84 nM T16117 D00EVC 10197851 IC50 = 100 nM T16117 D00KOE 18983431 IC50 = 10600 nM T16117 D00PEC 1331 Ki = 250 nM T16117 D00TDJ 44430622 IC50 = 4600 nM T16117 D01EHS 15552206 IC50 = 1000 nM T16117 D01ILO 15689 Ki = 410 nM T16117 D01MEA 22617750 IC50 = 1200 nM T16117 D01RGM 3311 Ki = 320 nM T16117 D01TDG 347590 Ki = 120 nM T16117 D01XOR 44396191 IC50 = 2700 nM T16117 D01YNT 10012278 IC50 = 3390 nM T16117 D02ELA 107984 Ki = 230 nM T16117 D02EOF 10725313 IC50 = 2600 nM T16117 D02MFQ 10606829 IC50 = 6800 nM T16117 D02OAB 761929 IC50 = 72000 nM T16117 D02TMX 9855524 IC50 = 10 nM T16117 D02TYS 44396204 IC50 = 2800 nM T16117 D02UKY 135415975 IC50 = 180000 nM T16117 D03CAJ 10375155 IC50 = 339 nM T16117 D03FJM 10198326 IC50 = 500 nM T16117 D03JXX 10261068 IC50 = 130 nM T16117 D03ODQ 15463448 IC50 = 17740 nM T16117 D03QMU 10104379 IC50 = 850 nM T16117 D03QSQ 19049087 IC50 = 17300 nM T16117 D03UTI 24728219 IC50 = 17000 nM T16117 D03WOZ 1893 IC50 = 2500 nM T16117 D04KUP 17842471 IC50 = 4300 nM T16117 D04PBI 44593548 Ki = 3000 nM T16117 D04QFO 44393534 IC50 = 9900 nM T16117 D05APC 19049123 IC50 = 390 nM T16117 D05VAB 9886249 IC50 = 741.31 nM T16117 D06VYU 10198539 IC50 = 440 nM T16117 D07BLJ 44322961 IC50 = 21000 nM T16117 D07GEN 393037 IC50 = 44000 nM T16117 D07INO 18428457 IC50 = 660 nM T16117 D07MFH 44323014 IC50 = 8390 nM T16117 D07OQX 9812839 IC50 = 13200 nM T16117 D07OVY 21894739 IC50 = 37000 nM T16117 D07PYV 10439 IC50 = 4800 nM T16117 D07VFC 42625451 IC50 = 490 nM T16117 D08ALG 9793728 IC50 = 3500 nM T16117 D08CMQ 18721725 IC50 = 1900 nM T16117 D08FXW 42625617 IC50 = 514 nM T16117 D08ISP 19049152 IC50 = 27000 nM T16117 D08JSR 3287412 IC50 = 17000 nM T16117 D08PZX 15463450 IC50 = 7100 nM T16117 D08UQH 53600 Ki = 105000 nM T16117 D08WEI 18721726 IC50 = 1800 nM T16117 D09BKV 15463449 IC50 = 2800 nM T16117 D09NRX 18721724 IC50 = 590 nM T16117 D0A6RU 11116249 IC50 = 4200 nM T16117 D0AO5D 1433 Ki = 2000 nM T16117 D0C1OB 12778904 IC50 = 20000 nM T16117 D0D0TO 85237 IC50 = 1100 nM T16117 D0D2WC 17892465 IC50 = 2400 nM T16117 D0D3CJ 10308091 IC50 = 13803.84 nM T16117 D0D4US 22352548 IC50 = 2400 nM T16117 D0D7PK 3268009 IC50 = 200 nM T16117 D0D9LT 12778906 IC50 = 3100 nM T16117 D0G4ZL 19049163 IC50 = 610 nM T16117 D0GX7G 5289555 Ki = 5300 nM T16117 D0H6JC 81829 IC50 > 1000000 nM T16117 D0I3ZP 44396203 IC50 = 160 nM T16117 D0I7VD 5139 Ki = 29 nM T16117 D0IR4Y 9995251 IC50 = 932 nM T16117 D0J1LO 445319 Ki = 37 nM T16117 D0J2RI 19049061 IC50 = 610 nM T16117 D0J7NS 15887953 IC50 = 800 nM T16117 D0K1CM 10749191 IC50 = 10000 nM T16117 D0K4SV 4102304 IC50 = 4900 nM T16117 D0K4YY 44399940 IC50 = 530 nM T16117 D0L9SL 44322997 IC50 = 25900 nM T16117 D0LB9U 44322572 IC50 = 6240 nM T16117 D0LE6N 19049158 IC50 = 310 nM T16117 D0LL3D 20323899 IC50 = 14000 nM T16117 D0M4BM 23042899 IC50 = 3700 nM T16117 D0N3HU 15463447 IC50 = 6800 nM T16117 D0N8EU 173566 IC50 = 10000 nM T16117 D0O3XZ 1533 IC50 = 40 nM T16117 D0O9II 189081 IC50 = 3200 nM T16117 D0OW8M 9797857 IC50 = 6000 nM T16117 D0R9KX 44399941 IC50 = 246 nM T16117 D0SB5H 18721719 IC50 = 830 nM T16117 D0T9ZQ 69681 IC50 = 59000 nM T16117 D0VB2W 21501 IC50 = 47000 nM T16117 D0VN7G 44393480 IC50 = 9600 nM T16117 D0W0OJ 417524 IC50 = 22000 nM T16117 D0W9UV 21507 IC50 = 98 nM T16117 D0X2XQ 10467406 IC50 = 1400 nM T16117 D0X5QJ 1649 IC50 = 170 nM T16117 D0X6MB 9942127 IC50 = 900 nM T16117 D0X6QY 19049121 IC50 = 140 nM T16117 D0XJ1C 10396852 IC50 = 80 nM T16117 D0Y0FS 24239 IC50 = 32000 nM T16117 D0Y2AO 2155 Ki = 12000 nM T98198 D0E3TC 44259 IC50 = 13.9 nM T98198 CP04JC 11666231 IC50 = 157 nM T98198 CV63UL 67240318 IC50 > 10000 nM T98198 CVIA91 71553085 IC50 = 8270 nM T98198 C1TR3O 71553152 IC50 = 24860 nM T98198 C2MD1Q 155513187 IC50 > 10000 nM T98198 D0N4LR 53469448 IC50 = 701 nM T98198 D0O6OH 71553154 IC50 = 4860 nM T85944 D08FKL 71466517 IC50 = 0.02 nM T85944 CWD65K 9906881 IC50 = 350 nM T85944 CR8NA2 10041662 IC50 = 160 nM T85944 C1QE2G 10090784 IC50 = 190 nM T85944 CGU29K 10427696 IC50 = 120 nM T85944 C09FXA 10858308 IC50 = 1600 nM T85944 C9B2RG 10871279 IC50 = 5500 nM T85944 CW34DT 10873013 IC50 = 9600 nM T85944 C3XZ0Y 10922966 IC50 = 5400 nM T85944 CMD4A8 10935650 IC50 = 21200 nM T85944 CLQ7O4 10956876 IC50 = 1400 nM T85944 CH6JG0 11044318 IC50 = 2700 nM T85944 CDE21T 11128226 IC50 > 50000 nM T85944 CG57AI 11128407 IC50 = 62500 nM T85944 CX5HQ0 11140377 IC50 = 31200 nM T85944 CSDO30 11546620 IC50 < 2.05 nM T85944 C6YJ3H 11811302 IC50 = 7400 nM T85944 C1CEL4 11822908 IC50 = 21700 nM T85944 CD13UQ 44336034 IC50 = 9000 nM T85944 CJ4SA0 44336181 IC50 = 6000 nM T85944 C8QME5 44336182 IC50 = 5500 nM T85944 C9MQ7Y 44336190 IC50 = 250 nM T85944 C6LAJ5 44336191 IC50 = 46000 nM T85944 C95QSX 44336199 IC50 = 1300 nM T85944 CWG8L5 44336202 IC50 = 38500 nM T85944 CY9AB2 44336206 IC50 = 500 nM T85944 CL0J8C 44336211 IC50 > 50000 nM T85944 C1TWP3 44336212 IC50 = 300 nM T85944 C5V1CT 44336221 IC50 = 1200 nM T85944 CTJW98 44336225 IC50 = 17800 nM T85944 CC0Q6W 44336244 IC50 = 840 nM T85944 C7FRN0 44336247 IC50 = 4900 nM T85944 CW2IC9 44336248 IC50 = 58700 nM T85944 C0L1QZ 44336275 IC50 = 18000 nM T85944 C0AC1K 44336302 IC50 > 60000 nM T85944 C2W5BF 44336325 IC50 = 960 nM T85944 CND26X 44336327 IC50 = 560 nM T85944 CVBG59 44336328 IC50 = 10000 nM T85944 C95YZR 44336334 IC50 > 30000 nM T85944 CR1VS2 44336335 IC50 > 30000 nM T85944 CQ1YZ4 44336337 IC50 > 50000 nM T85944 CR53ZM 44336338 IC50 = 7500 nM T85944 C7FD5R 44336339 IC50 = 1540 nM T85944 CZ29JG 44336341 IC50 = 12000 nM T85944 CUP68O 44336345 IC50 > 30000 nM T85944 CHK1G5 44336353 IC50 = 6000 nM T85944 CK3ZX4 44336359 IC50 > 50000 nM T85944 C6CR5P 44336372 IC50 = 20000 nM T85944 C8M9QB 44336373 IC50 = 3900 nM T85944 CHR9F7 44336376 IC50 = 7300 nM T85944 C2OV9Q 44336377 IC50 > 10000 nM T85944 CBW8G0 44336378 IC50 = 2500 nM T85944 CJ93OS 44336386 IC50 = 280 nM T85944 C0YLK1 44336388 IC50 = 7800 nM T85944 CPQE91 44336389 IC50 > 30000 nM T85944 C6QG8T 44336392 IC50 = 25000 nM T85944 COK8H6 44336396 IC50 = 5600 nM T85944 CM3YH9 44336397 IC50 = 10000 nM T85944 CVL0A9 44336400 IC50 = 2200 nM T85944 C03MKX 44336408 IC50 = 4900 nM T85944 C2JSG0 44336416 IC50 = 1000 nM T85944 CWED59 44336440 IC50 = 30000 nM T85944 CDB9O7 44336442 IC50 = 1000 nM T85944 CIST03 44336454 IC50 = 3300 nM T85944 CR8D7O 44336508 IC50 = 5000 nM T85944 C7JUG0 44427160 IC50 = 13000 nM T85944 C4BQI8 45137173 IC50 = 0.12 ug.mL-1 T85944 C2X3PO 45137174 IC50 = 0.014 ug.mL-1 T85944 CL79AZ 45254637 IC50 = 72 nM T85944 CT2QM0 45254832 IC50 = 3 nM T85944 CCK2F1 45254834 IC50 = 26 nM T85944 C0S2RG 45255036 IC50 = 4 nM T85944 CX95QA 46182721 IC50 = 0.004 ug.mL-1 T85944 CJ1D5H 51355299 IC50 = 49 nM T85944 C76EBD 51355300 IC50 = 13 nM T85944 CU2SX3 51355576 IC50 = 1.37 nM T85944 C0RKB9 51356116 IC50 = 21.6 nM T85944 CY5C7R 53247212 IC50 = 0.53 nM T85944 CR4FP9 53247213 IC50 = 0.52 nM T85944 CEKV98 53247214 IC50 = 1.5 nM T85944 C6S9MO 54754548 IC50 < 2.13 nM T85944 C5A9BQ 56593152 IC50 = 3.6 nM T85944 CB14TG 56950327 IC50 = 13.8 nM T85944 CQG1A6 56950462 IC50 > 67.9 nM T85944 CGD21Q 56950464 IC50 > 92.5 nM T85944 CB64IK 56950466 IC50 = 9.04 nM T85944 C56GZP 56950467 IC50 = 1.36 nM T85944 CAG56D 56950600 IC50 = 7.04 nM T85944 C8OF5L 56950601 IC50 = 26.1 nM T85944 C5NL7X 56950602 IC50 > 100 nM T85944 C6WO7M 56950603 IC50 = 3.54 nM T85944 C6TJD9 56950604 IC50 = 6.78 nM T85944 C2NY8A 56950605 IC50 = 22.1 nM T85944 CAS63K 56950606 IC50 = 27.8 nM T85944 CN0F4L 56950732 IC50 < 1.05 nM T85944 C2A9BC 56950733 IC50 = 1.74 nM T85944 CE62SM 56950734 IC50 = 0.64 nM T85944 CWZ35K 56950735 IC50 < 2.47 nM T85944 CR5TI7 56950736 IC50 = 29.7 nM T85944 CE57JS 56950737 IC50 = 73.6 nM T85944 CD3MV5 56950738 IC50 = 21.2 nM T85944 CYU45M 56950873 IC50 = 12.9 nM T85944 C3EK5W 56950874 IC50 = 12.7 nM T85944 CFSE62 56950875 IC50 = 9.49 nM T85944 C6YZ1P 56950876 IC50 = 1.2 nM T85944 CG1T5Z 56950877 IC50 = 3.68 nM T85944 C9KI6P 56950998 IC50 > 92.5 nM T85944 CN3CA9 56950999 IC50 = 1.85 nM T85944 CJ9YX4 56951000 IC50 = 11.9 nM T85944 CNAI20 56951002 IC50 = 31.4 nM T85944 CN54SJ 56951004 IC50 = 5.16 nM T85944 C49HGY 56951127 IC50 > 100 nM T85944 CJNX18 56951128 IC50 = 10.1 nM T85944 C9DGM2 56951130 IC50 = 92.7 nM T85944 CRY69J 56951133 IC50 = 30.4 nM T85944 C31RYW 56951251 IC50 > 100 nM T85944 C8KJ3F 56951254 IC50 > 95.2 nM T85944 CER8N9 56964907 IC50 = 1.1 nM T85944 CV05SA 57325599 IC50 = 4.4 nM T85944 C2L0KF 57325600 IC50 > 87 nM T85944 C08WNR 57325601 IC50 = 5.3 nM T85944 CAN7W6 57325602 IC50 = 12 nM T85944 CSOT04 57325603 IC50 = 3.7 nM T85944 CM5OT1 57325604 IC50 = 2.6 nM T85944 C3J4MI 57325605 IC50 = 1.8 nM T85944 CU3K6Y 57325689 IC50 = 2 nM T85944 CIO64H 57325690 IC50 = 1 nM T85944 C71GEC 57325770 IC50 = 1.2 nM T85944 CQ9D3L 57325771 IC50 = 1.3 nM T85944 CU7R0N 57325772 IC50 = 1.2 nM T85944 CY14ZD 57325773 IC50 = 2 nM T85944 C56CGV 57325774 IC50 = 1.2 nM T85944 CWF9S6 57325856 IC50 = 1.1 nM T85944 CC51LG 57325857 IC50 = 1.1 nM T85944 CY1Q7P 57326596 IC50 = 69 nM T85944 C6DN2Q 57326597 IC50 = 6 nM T85944 CFR2P7 57326598 IC50 = 6.7 nM T85944 C0N9YW 57326599 IC50 = 30 nM T85944 CN40JR 57326692 IC50 = 22 nM T85944 CKD5W6 57326693 IC50 = 4.9 nM T85944 C8E7NR 57326694 IC50 = 2.3 nM T85944 CD6B9P 57326695 IC50 = 57 nM T85944 C72RQV 57326696 IC50 = 8.5 nM T85944 CBSZ49 57326697 IC50 > 72 nM T85944 CH5X7W 57326793 IC50 > 100 nM T85944 C7O5NC 57326794 IC50 = 53 nM T85944 CC26HU 57326798 IC50 = 11 nM T85944 C7DGC8 57326892 IC50 = 60 nM T85944 C60JEW 57326893 IC50 > 100 nM T85944 C6V1PE 57326894 IC50 = 39 nM T85944 CBZ96S 57326895 IC50 = 6.4 nM T85944 C6T0FE 57326896 IC50 > 100 nM T85944 C1T7RH 57326898 IC50 = 4.1 nM T85944 C3SBD4 57326985 IC50 = 1.8 nM T85944 CVPY26 57326986 IC50 = 3.2 nM T85944 CZ4JV0 57326987 IC50 = 2.2 nM T85944 CAUQ23 57326988 IC50 = 3 nM T85944 C8AVE9 57326989 IC50 = 2.9 nM T85944 CQ4T2C 57326990 IC50 = 4.8 nM T85944 COY8P0 57326991 IC50 = 3.9 nM T85944 C1MB4Q 59323957 IC50 = 0.001 ug.mL-1 T85944 CZBK04 59323986 IC50 = 0.006 ug.mL-1 T85944 C2U3LR 59324040 IC50 = 0.026 ug.mL-1 T85944 C4C5MB 59324049 IC50 = 0.3 ug.mL-1 T85944 CYGQ49 59697043 IC50 = 8 nM T85944 CEL13R 59697134 IC50 = 0.0005 ug.mL-1 T85944 COFJ15 59697419 IC50 = 20 nM T85944 CK0F2C 59697564 IC50 = 0.0012 ug.mL-1 T85944 C6V2GZ 70681060 IC50 = 390 nM T85944 CUV1Z4 70681061 IC50 = 160 nM T85944 CBV7G4 70683179 IC50 = 286 nM T85944 CE4Y1N 70685260 IC50 = 0.8 nM T85944 CYJ4O2 70687411 IC50 = 0.4 nM T85944 CC5E8F 70687412 IC50 = 0.4 nM T85944 CI7EP8 70689467 IC50 = 22 nM T85944 CF27TD 70689468 IC50 = 28 nM T85944 CKJR81 70689469 IC50 = 15 nM T85944 C2UXL6 70691578 IC50 = 3.3 nM T85944 CS95XK 70691579 IC50 = 3 nM T85944 C2PD4Y 70693659 IC50 = 8 nM T85944 CKWS13 70693660 IC50 = 90 nM T85944 CI1XN4 70693661 IC50 = 51 nM T85944 CULZ56 70693662 IC50 = 18 nM T85944 CQ4A7L 70693663 IC50 = 0.8 nM T85944 C7QX6F 70693664 IC50 = 0.376 nM T85944 C2KNR7 70693665 IC50 = 0.6 nM T85944 CTAP76 70695775 IC50 = 25 nM T85944 CJD06P 70695776 IC50 = 311 nM T85944 C1V8KM 86287507 IC50 = 4400 nM T85944 CD6NB0 89072105 IC50 = 0.083 ug.mL-1 T85944 CN1F9W 118721344 IC50 = 8700 nM T85944 CO43QG 118721345 IC50 = 14000 nM T85944 CO4N1K 118721346 IC50 = 92000 nM T85944 CY6K5B 118721347 IC50 = 33000 nM T85944 C2ZUC0 118721348 IC50 = 139000 nM T85944 CHXO25 118721349 IC50 = 3000 nM T85944 C0XWD1 118721350 IC50 = 7500 nM T85944 CH7ML9 118721351 IC50 = 2700 nM T85944 CS2OY3 118721352 IC50 = 2600 nM T85944 CT6WY0 118721353 IC50 = 5800 nM T85944 CAFU13 118721634 IC50 = 10000 nM T85944 CY9BP8 118721635 IC50 = 6100 nM T85944 C7S9NJ 118721636 IC50 = 2000 nM T85944 C0TG8I 118721637 IC50 = 1700 nM T85944 CY2LJ3 118721638 IC50 = 200 nM T85944 C3U0NC 118721639 IC50 = 3100 nM T85944 C40SZF 118721640 IC50 = 82500 nM T85944 C8NVJ6 118721641 IC50 = 8600 nM T85944 C7SV3Z 136110969 IC50 > 30000 nM T85944 CZFW82 137631443 IC50 = 3 nM T85944 CI1A0V 137633969 IC50 = 18 nM T85944 C3MAI2 137635134 IC50 = 8 nM T85944 CIAN30 137635731 IC50 = 0.002 ug.mL-1 T85944 C6VCP0 137636280 IC50 = 0.12 ug.mL-1 T85944 CR06JX 137636822 IC50 = 0.4 nM T85944 C2C1BR 137636869 IC50 = 14 nM T85944 C5N4EQ 137638052 IC50 = 8 nM T85944 CM68HB 137638519 IC50 = 2 nM T85944 CBC3W7 137639716 IC50 = 13 nM T85944 CD0JK9 137639783 IC50 = 0.041 ug.mL-1 T85944 C6OAB5 137640599 IC50 = 0.035 ug.mL-1 T85944 C6THB1 137643027 IC50 = 63 nM T85944 CHRM65 137643088 IC50 = 0.002 ug.mL-1 T85944 C34CRT 137643862 IC50 = 14 nM T85944 C2OR6T 137645072 IC50 = 5 nM T85944 CF30YJ 137645503 IC50 = 4 nM T85944 C3RKI5 137645839 IC50 = 1 nM T85944 CYXC37 137646968 IC50 = 0.0004 ug.mL-1 T85944 CA68FK 137648995 IC50 = 108 nM T85944 CM3LT6 137649296 IC50 = 616 nM T85944 C69JFH 137649541 IC50 = 214 nM T85944 CV6BG5 137649553 IC50 = 20 nM T85944 C37EVR 137650278 IC50 = 6 nM T85944 CZ01VA 137651154 IC50 = 72 nM T85944 CYP2B7 137651506 IC50 = 6 nM T85944 CY8B2O 137651547 IC50 = 0.005 ug.mL-1 T85944 C4KG2Q 137653077 IC50 = 30 nM T85944 CTZS78 137653870 IC50 = 26 nM T85944 CPN08E 137654857 IC50 = 0.011 ug.mL-1 T85944 CIW0S1 137654906 IC50 = 2 nM T85944 CIM5Q1 137655566 IC50 = 5 nM T85944 CLB60K 137656147 IC50 = 4 nM T85944 C1O8DB 137657296 IC50 = 333 nM T85944 CX5LN7 137657576 IC50 = 15 nM T85944 C8L3KH 137658300 IC50 = 10 nM T85944 CDBV75 137658829 IC50 = 0.53 ug.mL-1 T85944 CMB7C1 137659259 IC50 = 14 nM T85944 CQK4E7 137660427 IC50 = 2 nM T85944 C34LEF 137661409 IC50 = 5 nM T85944 CVWB64 137661442 IC50 = 50 nM T85944 CP3FA0 137661749 IC50 = 6 nM T37961 D0D9JW 3826 IC50 = 36000 nM T37961 D06YWH 11178236 IC50 = 500 nM T37961 D07SDQ 969516 IC50 = 16000 nM T37961 D08MHM 25227462 IC50 = 13.7 nM T37961 D0E3TC 44259 IC50 = 0.3 nM T37961 D0Q7RE 16007391 Ki > 10000 nM T37961 D0U3EP 445154 IC50 = 15000 nM T37961 CUQH50 79515 IC50 = 38000 nM T37961 CRB15U 521106 IC50 = 1000 nM T37961 CI87QT 756681 IC50 = 18000 nM T37961 C3J7LB 2951910 IC50 = 48.4 nM T37961 CO9C2V 3081033 IC50 = 2500 nM T37961 CNL8W2 4046054 IC50 = 23000 nM T37961 CR6N2P 5064557 IC50 = 23000 nM T37961 CBOP58 11293798 Ki > 10000 nM T37961 C26BZX 11362471 Ki > 10000 nM T37961 CWXB93 11397177 Ki > 10000 nM T37961 CTG83F 11539329 Ki > 9700 nM T37961 CACS26 11561968 Ki > 2000 nM T37961 CMIL86 11590363 Ki > 9700 nM T37961 CSM62L 11626920 IC50 > 30000 nM T37961 C9T6SC 11640926 Ki > 9700 nM T37961 CU0E8O 11690457 Ki > 2000 nM T37961 CU0M1E 11947684 IC50 < 1 nM T37961 C0ZWP3 15953852 Ki = 50 nM T37961 CFPW41 16007116 Ki > 9700 nM T37961 C1FC4H 21939235 Ki = 100 nM T37961 CE0RM2 23734191 IC50 = 31000 nM T37961 C7YG1N 24759534 IC50 = 8300 nM T37961 C6GC3X 25014511 IC50 = 3100 nM T37961 CY3HW5 46224684 IC50 = 510 nM T37961 CLS29B 46872626 IC50 > 10000 nM T37961 C2O8RZ 46886323 IC50 = 531 nM T37961 CN9QD7 56643097 IC50 > 10000 nM T37961 CXJ63M 59603829 IC50 = 6200 nM T37961 CQEU96 59603842 IC50 = 24 nM T37961 COH62U 60097413 IC50 > 10000 nM T37961 C1MR8Q 60097495 IC50 > 10000 nM T37961 CE12XV 60163664 Ki > 4500 nM T37961 C6DUK0 60163745 Ki > 4500 nM T37961 C8BV6Z 60163908 Ki > 4500 nM T37961 CDYE40 60164283 Ki > 4500 nM T37961 CCUH92 60164742 Ki > 4500 nM T37961 C4GK3V 60164846 Ki > 4500 nM T37961 CV63UL 67240318 IC50 > 10000 nM T37961 C12DPO 68060125 IC50 <= 10 nM T37961 C36BVQ 68181618 Ki > 4500 nM T37961 CUQ4F0 68181642 Ki > 4500 nM T37961 CAN7U2 68181681 Ki > 4500 nM T37961 CK7XJ5 68181838 Ki > 4500 nM T37961 CFQ9N0 68181876 Ki > 4500 nM T37961 C4VK1Q 68181882 Ki > 4500 nM T37961 CQC0R5 68181954 IC50 = 2000 nM T37961 C5DGR9 69036886 IC50 = 10000 nM T37961 C3GTU1 69762142 IC50 > 10000 nM T37961 C82YNL 70934541 IC50 = 7.7 nM T37961 CKT60L 71455860 Ki > 9700 nM T37961 CQA4U7 71528975 Ki = 4 nM T37961 CT7V2J 71529158 Ki = 6.75 nM T37961 CT94VL 71543346 IC50 = 4000 nM T37961 C83FVQ 71557891 IC50 <= 10 nM T37961 CRX81Q 71575642 IC50 > 10000 nM T37961 CH97AJ 71611283 Ki = 120 nM T37961 C3FLP7 71611421 Ki = 32 nM T37961 CZA4N8 71611423 IC50 = 685 nM T37961 CQ6I7D 71611843 Ki = 4 nM T37961 CUOV67 71713028 EC50 = 1510 nM T37961 C04YBD 71713176 EC50 = 4720 nM T37961 CLNT74 71713177 IC50 = 227 nM T37961 CAM0H8 71713178 IC50 = 487 nM T37961 C93CWH 71713179 EC50 = 2350 nM T37961 C74CZR 71713180 IC50 = 2140 nM T37961 CW5F6M 71713181 IC50 = 2680 nM T37961 C80ELC 71713328 IC50 = 5210 nM T37961 CI2K9F 71713330 IC50 = 4670 nM T37961 C4GS2T 71713331 EC50 = 17600 nM T37961 CTIL17 71713332 EC50 = 7990 nM T37961 C96EQU 71713333 EC50 = 3780 nM T37961 CC3AF0 71713471 IC50 = 2880 nM T37961 C0E2IY 71713472 IC50 = 11300 nM T37961 CCRH57 71713473 EC50 = 10900 nM T37961 CDIU43 71713474 EC50 = 27700 nM T37961 CD5XP1 71713475 EC50 = 61300 nM T37961 CX7U9Z 71713614 EC50 = 50100 nM T37961 C64BQO 71713615 EC50 = 39600 nM T37961 C79OKU 71713616 EC50 = 21300 nM T37961 C1XA9Y 71713617 IC50 = 126 nM T37961 CD94MY 71713618 IC50 = 61 nM T37961 CU1E5J 71713768 EC50 = 1040 nM T37961 CDNS94 71713769 EC50 = 3590 nM T37961 CPY19I 71720361 EC50 = 4730 nM T37961 C0DL3F 72698602 IC50 < 1 nM T37961 C0OPM4 72725813 Ki > 4500 nM T37961 CSN7R9 73347511 IC50 = 8360 nM T37961 C9YEQ2 73350469 Ki = 5.13 nM T37961 CF8LD4 73356518 Ki = 4.2 nM T37961 CWK65Y 76329224 Ki > 4500 nM T37961 C9M6JR 76332879 Ki = 15300 nM T37961 CJ2T9E 76332983 IC50 > 10000 nM T37961 C6Z5SJ 77232204 IC50 = 64 nM T37961 CUF60Q 86274945 IC50 > 4500 nM T37961 CA9G2O 86762626 Ki = 120 nM T37961 CK4P6C 89650573 Ki = 6 nM T37961 C2OAX6 89650963 Ki = 5 nM T37961 CAP3J9 89651542 Ki = 68 nM T37961 CH62LD 89658721 Ki = 84 nM T37961 C5Y4TD 89658723 Ki = 25 nM T37961 C87OKB 89658750 Ki = 18 nM T37961 C1HW4B 89735655 IC50 = 2100 nM T37961 C49LZW 89766055 Ki = 25 nM T37961 CS2A8K 90466181 Ki = 1.9 nM T37961 CC69QY 90467635 Ki = 6.1 nM T37961 CR9ZA2 90467636 Ki = 6 nM T37961 C6JE2B 90467771 Ki = 19 nM T37961 C29IOE 90468049 Ki = 2.1 nM T37961 CYHR27 91664373 Ki = 3.7 nM T37961 C1YKE5 91808045 IC50 = 323 nM T37961 C6Y4PV 91809512 Ki = 22 nM T37961 C8Y2GZ 91809513 Ki = 21 nM T37961 CDO9I1 101884431 IC50 = 14 nM T37961 CC9G8U 101884433 IC50 = 1 nM T37961 CR9GZ5 101884437 IC50 = 43 nM T37961 C3XJI0 101884438 IC50 = 48 nM T37961 COK7A6 117833359 Ki = 8 nM T37961 CP3LR1 117833406 Ki = 7.4 nM T37961 CVZ6A9 117833539 Ki = 1.9 nM T37961 CY61TV 117833566 Ki = 4.3 nM T37961 CIM4B7 118720596 IC50 > 4500 nM T37961 CQCX41 118737057 IC50 > 10000 nM T37961 C9VYJ0 119057464 Ki = 4.6 nM T37961 CQBV93 122164606 IC50 = 260 nM T37961 C9X4WQ 122178544 Ki = 179 nM T37961 C0HWD7 122178545 Ki = 33 nM T37961 C48HAL 122178546 Ki = 48 nM T37961 CB1KW7 122178547 Ki = 33 nM T37961 C5PKU2 122178548 Ki = 18 nM T37961 C01QJE 122178550 Ki = 119 nM T37961 C87ERY 122178551 Ki = 454 nM T37961 C30LEZ 122178552 Ki = 561 nM T37961 C4NSI0 122178553 Ki = 4390 nM T37961 C41KSU 122178554 Ki = 245 nM T37961 C3BHS9 122178555 Ki = 157 nM T37961 CDUA42 122182198 Ki = 16 nM T37961 C30URY 122182199 Ki = 29 nM T37961 CNZG96 122182482 Ki = 373 nM T37961 C9ENM4 122182483 Ki = 552 nM T37961 CV3X7Z 122182484 Ki = 18 nM T37961 CV7E8D 122182485 Ki = 111 nM T37961 CFP8L3 122182486 Ki = 37 nM T37961 C41VZY 122182487 Ki = 49 nM T37961 C9Z5AY 122182488 Ki = 362 nM T37961 CSN1P8 122182489 Ki = 18 nM T37961 C74VXS 122182490 Ki = 46 nM T37961 CL3PR1 122182491 Ki > 4500 nM T37961 CQ8XC0 122183105 IC50 = 83 nM T37961 C3C5DB 122183106 IC50 = 18 nM T37961 C4D6UX 122183107 IC50 = 460 nM T37961 C7GO9K 122183108 IC50 = 6300 nM T37961 C0FDH2 122183109 IC50 = 400 nM T37961 CHS65F 122183110 IC50 = 63 nM T37961 CJY0F1 122183111 IC50 = 120 nM T37961 C21BIY 122183112 IC50 = 740 nM T37961 C8J7MS 122183113 IC50 = 490 nM T37961 CGAY53 122183114 IC50 = 2000 nM T37961 C3IOU4 122183115 IC50 = 630 nM T37961 CR3VI7 122183116 IC50 = 84 nM T37961 C1DR5U 122183117 IC50 = 88 nM T37961 C31TRU 122183118 IC50 = 650 nM T37961 CDJ59L 122183119 IC50 = 13 nM T37961 CHPN18 122183120 IC50 = 7.5 nM T37961 C1XI4H 122183121 IC50 = 23 nM T37961 CT8E2Y 122183122 IC50 = 630 nM T37961 CE5ZP2 122183123 IC50 = 440 nM T37961 CF4IX9 122183124 IC50 = 7.6 nM T37961 CS4B8U 122183125 IC50 = 21 nM T37961 C92QGD 122183126 IC50 = 3 nM T37961 C95ZQH 122183127 IC50 = 12 nM T37961 C5Y8UJ 122183128 IC50 = 55 nM T37961 CD19ZM 122183129 IC50 = 37 nM T37961 CAE3H1 122183130 IC50 = 130 nM T37961 CEP9G6 122183131 IC50 = 140 nM T37961 CMO5R6 122183132 IC50 = 5.8 nM T37961 CPG4C1 122183133 IC50 = 33 nM T37961 C0ZFP1 122183134 IC50 = 4.5 nM T37961 CBL41Y 122183173 IC50 = 270 nM T37961 CH0LK7 122183174 IC50 = 2.8 nM T37961 C04VNA 122187536 IC50 = 900 nM T37961 C4X7SD 122192466 IC50 > 10000 nM T37961 C1U5KH 127028469 Ki = 64 nM T37961 C4EV0I 127028470 Ki = 66 nM T37961 CYF4L7 127029374 Ki = 7.9 nM T37961 C3SF4U 127048382 Ki = 5.9 nM T37961 C9ZC0R 127048383 Ki = 9 nM T37961 CUOQ15 127048384 Ki = 2.7 nM T37961 C9ZS6X 127048385 Ki = 4.4 nM T37961 CTJ50H 127048386 Ki = 0.95 nM T37961 CEL91I 127048725 Ki = 3.5 nM T37961 CGD90Y 127048726 Ki = 6.7 nM T37961 C94JNY 127048727 Ki = 8 nM T37961 CBP5T0 127048728 Ki = 6.3 nM T37961 CG5B3H 127048729 Ki = 17 nM T37961 C5FT0P 127049039 Ki = 56 nM T37961 CV8C5H 127049121 Ki = 360 nM T37961 CZL5T2 127049404 Ki = 3.3 nM T37961 CQO72D 127049720 Ki = 89 nM T37961 CLB7V2 127049721 Ki = 13 nM T37961 CJC5B2 127050025 Ki = 36 nM T37961 CDRB26 127050517 Ki = 11 nM T37961 CFO30S 127051514 Ki = 382 nM T37961 CZG30T 127051548 Ki = 950 nM T37961 CFQ18V 127051549 Ki = 943 nM T37961 C4P1UT 127052177 Ki = 11 nM T37961 C8AX0O 127052178 Ki = 5.2 nM T37961 CN37MB 127052179 Ki = 22 nM T37961 CE2B9V 127052180 Ki = 372 nM T37961 CT2RO3 127052399 Ki = 23 nM T37961 CQK91G 127052400 Ki = 119 nM T37961 CR6A5U 127053076 Ki = 13 nM T37961 C8F0DQ 129909860 IC50 < 1 nM T37961 CK6YP3 132274772 Ki > 10000 nM T37961 CJ9D8A 132274773 Ki > 10 nM T37961 CJ75FW 134132809 IC50 = 3 nM T37961 C9RZ3P 134134011 IC50 = 0.45 nM T37961 CPB92K 134137028 IC50 = 45 nM T37961 C90YTL 134137370 IC50 = 19 nM T37961 CQ07CH 134139098 IC50 = 2.8 nM T37961 CNOR21 134142020 IC50 = 2.1 nM T37961 CI6W3K 134142647 IC50 = 1.5 nM T37961 C0F3RD 134146595 IC50 = 2 nM T37961 CEU91D 134147801 IC50 = 0.35 nM T37961 C82HSO 134149733 IC50 = 33 nM T37961 C5RAG2 134150175 IC50 = 0.58 nM T37961 C15YCV 134151598 IC50 = 8.7 nM T37961 C74SCK 134154467 IC50 = 3300 nM T37961 CQLM73 134154799 IC50 = 14 nM T37961 CT29UB 134156831 IC50 = 9.6 nM T37961 C2AN7T 134611886 IC50 > 100000 nM T37961 C52FCI 134817245 Ki = 690 nM T37961 C5AK2R 135198771 Ki > 4520 nM T37961 CD85HP 135198778 Ki > 10000 nM T37961 CFI13G 135198787 Ki = 2750 nM T37961 CQUW03 135198795 Ki > 4520 nM T37961 CGJ4P7 135198796 Ki > 4520 nM T37961 C3AP4K 135198799 Ki = 368 nM T37961 CEML07 135199057 Ki = 2080 nM T37961 C8WSL3 135567021 IC50 = 18 nM T37961 C63FEC 137125241 IC50 = 5.2 nM T37961 CIHJ46 137125256 IC50 = 54000 nM T37961 CI81AE 137125257 IC50 = 190 nM T37961 CV6WC3 137348710 Ki = 3112 nM T37961 CNE1Y9 137631969 IC50 = 65 nM T37961 CGQZ93 137632703 Ki > 4520 nM T37961 C8S7YK 137634619 Ki = 383 nM T37961 C5S7PK 137635580 Ki = 503 nM T37961 C3X7SM 137641415 Ki = 2085 nM T37961 CAO28T 137644956 Ki = 1891 nM T37961 CXJQ26 137648567 Ki = 401 nM T37961 C1B4LS 137649300 Ki = 288 nM T37961 C8SV7X 137653128 Ki > 4520 nM T37961 CXK23M 137659630 Ki = 1072 nM T37961 C6VB3O 145925651 IC50 >= 5000 nM T37961 C25EGT 145987455 IC50 = 1000 nM T37961 C2MD1Q 155513187 IC50 > 10000 nM T37961 D00ERW 44444843 Ki > 9727 nM T37961 D00HVA 11624601 Ki > 9700 nM T37961 D07ORL 73348907 Ki = 36.8 nM T37961 D0L2WP 46225540 IC50 = 31 nM T37961 D0Q3NG 11715520 Ki > 9700 nM T37961 D0S3TJ 76098 IC50 = 18000 nM T37961 D0S7IE 11658882 Ki > 9700 nM T37961 D0U4VL 5472440 IC50 = 25000 nM T93783 D0E3SH 6918837 EC50 = 130 nM T93783 D0E7PQ 5311 EC50 = 2300 nM T93783 C0ZS7W 1570036 EC50 > 40000 nM T93783 C0I4VB 1582691 EC50 = 6700 nM T93783 CJYF70 2055715 EC50 > 40000 nM T93783 CX8ZD5 2480904 EC50 > 40000 nM T93783 C4Q0LV 2673048 EC50 = 24000 nM T93783 CR2I9T 2673049 EC50 = 13000 nM T93783 C5MY7U 2673051 EC50 > 40000 nM T93783 CQP38X 2673140 EC50 > 40000 nM T93783 COT82Z 2678134 EC50 > 40000 nM T93783 C4LCS2 2679227 EC50 > 40000 nM T93783 C1R9FI 3148065 EC50 > 40000 nM T93783 CF1ZX9 3148068 EC50 > 40000 nM T93783 CDP65B 3392495 EC50 > 40000 nM T93783 CJ32NW 5276854 EC50 = 10000 nM T93783 C1X8CH 8919483 EC50 = 1700 nM T93783 CL14MN 11228475 IC50 = 19000 nM T93783 CU0M1E 11947684 EC50 = 220 nM T93783 CQFH26 16657874 EC50 = 1000 nM T93783 CL0ZG8 26197793 EC50 > 40000 nM T93783 CRBJ58 29985358 EC50 > 40000 nM T93783 C5KS8P 31845722 EC50 > 40000 nM T93783 CZ0W8P 35023502 EC50 = 20000 nM T93783 C9AQ2B 44476170 IC50 = 6000 nM T93783 C23VQS 44538018 IC50 = 10000 nM T93783 C0IUO1 44538110 IC50 = 30000 nM T93783 C9L6GY 46878878 IC50 = 7000 nM T93783 CC79KB 46878886 IC50 = 12000 nM T93783 C15AUN 46878888 IC50 = 35000 nM T93783 CVC6D7 46878889 IC50 = 16000 nM T93783 C51ICG 46878890 IC50 = 900 nM T93783 C6B7WU 47149286 EC50 = 19000 nM T93783 C95CET 47267102 EC50 > 40000 nM T93783 C0S4DV 49317486 EC50 > 40000 nM T93783 C98BLM 49871817 EC50 = 8100 nM T93783 CI0C1T 84330289 EC50 > 40000 nM T93783 CUW59A 84353474 EC50 = 13000 nM T93783 C8FH5C 84376194 EC50 = 8000 nM T93783 CA25LU 84581125 EC50 > 40000 nM T93783 C9VW6E 145420081 EC50 = 4700 nM T93783 CBU1J2 145420084 EC50 = 5000 nM T93783 CVY72T 145420089 EC50 > 40000 nM T93783 CN4O1E 145420093 EC50 = 11000 nM T93783 CFHJ67 145420094 EC50 > 40000 nM T93783 CK73BX 145420104 EC50 = 1200 nM T93783 C24LCH 145420105 EC50 = 2700 nM T93783 CAP58Q 145420115 EC50 > 40000 nM T93783 CS7IX9 145420121 EC50 > 40000 nM T93783 C2M0AP 145420133 EC50 > 40000 nM T93783 CZ3E9Y 145420134 EC50 = 1300 nM T93783 C0OKY9 145420135 EC50 = 4300 nM T93783 CRSJ29 145420136 EC50 = 3600 nM T93783 CT3R4Q 145420139 EC50 = 3700 nM T93783 C9KL0H 145420152 EC50 = 2900 nM T93783 C1Q6UK 145420161 EC50 > 40000 nM T93783 CB4JK2 145420162 EC50 = 13000 nM T93783 CE0NG8 145420163 EC50 = 6400 nM T93783 CVND14 145420166 EC50 = 1900 nM T93783 CA8G0Q 145420168 EC50 = 2600 nM T93783 C0JE3D 145420172 EC50 > 40000 nM T93783 CE48UV 145420175 EC50 = 2600 nM T93783 CXRV29 145420176 EC50 = 3600 nM T93783 CCX28B 145420182 EC50 = 1500 nM T93783 CGB0S1 145420184 EC50 = 6300 nM T93783 C8PV1N 145420185 EC50 = 9200 nM T93783 CN0Q7K 146227891 EC50 = 6400 nM T93783 CE36BL 155510895 EC50 = 4700 nM T93783 CMCN18 155513932 EC50 = 3300 nM T93783 COS61G 155518226 EC50 = 2900 nM T93783 CB32WT 155518767 EC50 = 900 nM T93783 CHX85M 155518985 EC50 = 23000 nM T93783 CK0GR8 155521142 EC50 = 1300 nM T93783 C0FK3S 155521424 EC50 > 40000 nM T93783 CUPV38 155521580 EC50 > 40000 nM T93783 CZ3DU8 155523431 EC50 > 40000 nM T93783 CC50XQ 155523517 EC50 > 40000 nM T93783 CR0EG6 155523860 EC50 > 40000 nM T93783 CDH0S3 155525311 EC50 > 40000 nM T93783 CU4NW9 155525612 EC50 > 40000 nM T93783 CR6PL3 155525929 EC50 = 2800 nM T93783 C16ETJ 155525958 EC50 > 40000 nM T93783 CBU3E9 155528001 EC50 = 3100 nM T93783 C5IRS7 155530014 EC50 = 2300 nM T93783 CY8M3G 155530940 EC50 = 2700 nM T93783 CPN3D5 155531584 EC50 > 40000 nM T93783 CG8U4C 155532355 EC50 > 40000 nM T93783 CD6L2W 155535495 EC50 > 40000 nM T93783 CVIN48 155541359 EC50 > 40000 nM T93783 CANX75 155541646 EC50 = 22000 nM T93783 CT58ZW 155542993 EC50 = 4700 nM T93783 CF19EA 155543343 EC50 > 40000 nM T93783 COF3U6 155543987 EC50 = 800 nM T93783 C30WGE 155544176 EC50 > 40000 nM T93783 CWVA75 155545969 EC50 = 1400 nM T93783 CU93RH 155546257 EC50 = 3700 nM T93783 C3DE4Y 155547004 EC50 = 40000 nM T93783 CZDT05 155547368 EC50 > 40000 nM T93783 CCJ98Y 155549173 EC50 > 40000 nM T93783 C4KIG5 155549469 EC50 > 40000 nM T93783 CU5ED2 155549471 EC50 = 11000 nM T93783 C58RLJ 155549712 EC50 = 2200 nM T93783 CSN34H 155551296 EC50 > 40000 nM T93783 CME4B8 155551437 EC50 > 40000 nM T93783 CV80GB 155551552 EC50 > 40000 nM T93783 C7S2AP 155552810 EC50 > 40000 nM T93783 CAR32L 155553594 EC50 = 4700 nM T93783 CFY6J7 155553849 EC50 = 3000 nM T93783 C9RQ5D 155554505 EC50 > 40000 nM T93783 CBJ57Z 155556288 EC50 > 40000 nM T93783 CB18ZI 155556851 EC50 > 40000 nM T93783 CUH9N4 155559369 EC50 > 40000 nM T93783 CVQ5R4 155559643 EC50 > 40000 nM T93783 CT90CG 155560622 EC50 > 40000 nM T93783 CUBY52 155562312 EC50 = 11000 nM T93783 CZO7A1 155565161 EC50 > 40000 nM T93783 CPV46I 155567368 EC50 > 40000 nM T13644 D0TV0C 9941444 Ki = 0.7943 nM T13644 D06JFI 11251755 EC50 = 3.33 nM T13644 D0J8PI 158782 IC50 = 880 nM T13644 D09JXL 5311430 Ki = 31.62 nM T13644 D0Y2HR 2247 Ki > 10000 nM T13644 C7V5WO 3156873 Ki = 2337 nM T13644 C6XYL5 6918011 Ki = 63.1 nM T13644 CHM63P 6918026 Ki = 19.95 nM T13644 CN20OR 9802240 Ki = 60 nM T13644 C63PHY 9803491 Ki = 430 nM T13644 C8SK1I 9803492 Ki = 3800 nM T13644 CR0U6E 9827283 Ki = 2574 nM T13644 CA8UQ7 9848232 Ki = 5686 nM T13644 CW3TM5 9851998 Ki = 2660 nM T13644 CTRI07 9852911 Ki = 2800 nM T13644 C9BJ3Q 9854636 IC50 = 750 nM T13644 CMLP16 9918828 Ki = 125.89 nM T13644 C3Z5YJ 9963342 Ki = 0.7943 nM T13644 CIT57N 9985523 Ki = 3300 nM T13644 C64LIB 10009650 Ki = 900 nM T13644 C58EOI 10053855 Ki > 10000 nM T13644 CL6G0Z 10094509 Ki = 36 nM T13644 C9C7RK 10096510 Ki = 3700 nM T13644 CFZN71 10166743 Ki = 79 nM T13644 CI21CK 10179247 Ki = 210 nM T13644 C6DRE9 10210016 Ki = 200 nM T13644 C4M9GN 10248767 Ki = 2500 nM T13644 CSY5K2 10325243 Ki = 3000 nM T13644 CL87OB 10411795 Ki = 170 nM T13644 CS96ON 10534086 IC50 = 140 nM T13644 CHZ9I8 10554930 Ki = 6200 nM T13644 CY3ZE9 10577746 IC50 = 3090 nM T13644 C9C0HF 10580397 Ki = 600 nM T13644 CU3DQ6 10630127 Ki = 93 nM T13644 C45JIZ 10699714 Ki = 6400 nM T13644 CG2UX4 10701257 IC50 = 934 nM T13644 CP0F7C 10724811 IC50 = 1380 nM T13644 CJM47E 10748701 IC50 = 733 nM T13644 CWF2N5 10748831 IC50 = 68 nM T13644 CLW4V6 10770814 Ki = 3300 nM T13644 CO56HI 10772403 IC50 = 1361 nM T13644 CGN0Z5 10772578 IC50 = 373 nM T13644 C3L4DH 10796238 IC50 = 1000 nM T13644 C15QGO 10819673 IC50 = 1000 nM T13644 CFL71O 10843862 IC50 = 216 nM T13644 C2PJ1O 10876898 Ki = 1.995 nM T13644 C35OXW 10917657 Ki = 6.9 nM T13644 C2CXF3 10960879 Ki = 71 nM T13644 C6TVQ8 10964197 Ki = 19.95 nM T13644 CXDG12 10996788 Ki = 0.3162 nM T13644 COU1Q7 11025614 Ki = 750 nM T13644 C4SCO8 11048825 Ki = 3.4 nM T13644 C1CD0X 11049745 Ki = 17 nM T13644 C56YON 11069321 IC50 = 0.8 nM T13644 C6AW0M 11112736 Ki = 0.64 nM T13644 CK1RX4 11136828 Ki = 1.585 nM T13644 CR1JP9 11147505 Ki = 0.7943 nM T13644 C1I9EX 11159133 IC50 = 587 nM T13644 C7REL4 11170698 IC50 = 35.7 nM T13644 CIEM12 11170867 IC50 > 1000 nM T13644 CW2JA8 11182381 IC50 = 18 nM T13644 CE3GC2 11205475 EC50 = 4.7 nM T13644 CXI32T 11205496 IC50 = 271 nM T13644 C2RNJ5 11205515 IC50 = 247 nM T13644 CUT8Z0 11240205 IC50 = 330 nM T13644 CK78SD 11240206 IC50 = 22 nM T13644 C67WXD 11274767 IC50 = 8.2 nM T13644 COK06N 11320738 IC50 = 600 nM T13644 C5D6AM 11332138 IC50 = 897 nM T13644 C5PAN4 11343811 IC50 = 623 nM T13644 CLQ53A 11355270 IC50 = 664 nM T13644 CQ0UC7 11378229 EC50 = 0.53 nM T13644 CC09ZU 11378299 IC50 = 624 nM T13644 CG7PT9 11389178 IC50 = 780 nM T13644 CFJD72 11423410 IC50 = 347 nM T13644 C4S2HG 11434734 IC50 = 53 nM T13644 C6XHC3 11457491 IC50 > 1000 nM T13644 CJ5A9B 11457521 IC50 = 650 nM T13644 CMA8C7 11468709 IC50 > 1000 nM T13644 CG8A0J 11468887 IC50 = 10 nM T13644 CZ3N5J 11468916 IC50 = 16 nM T13644 CORY59 11480246 IC50 = 14 nM T13644 C63QMX 11535351 IC50 > 1000 nM T13644 CF6K7M 11563877 IC50 = 360 nM T13644 CS68YA 11642413 IC50 = 6330 nM T13644 CZHN61 11678313 IC50 = 430 nM T13644 CW65KY 11705763 Ki = 170 nM T13644 CN63YV 11787877 IC50 > 1000 nM T13644 CR6UF9 11788180 IC50 = 1025 nM T13644 CK4U8N 11804376 IC50 = 648 nM T13644 C9XH7F 11815114 Ki = 0.631 nM T13644 CRA01O 11845058 IC50 = 210 nM T13644 C8X3CL 11845059 IC50 = 958 nM T13644 CO3HT9 11847587 IC50 = 942 nM T13644 CAD8P9 11848624 Ki > 10000 nM T13644 CM49QW 11848625 Ki > 10000 nM T13644 CEBA46 11848626 Ki > 10000 nM T13644 CCT5G7 11848677 Ki > 10000 nM T13644 CMR10F 11848679 Ki > 10000 nM T13644 C9QDX3 11848833 Ki > 10000 nM T13644 CL6B5X 11848835 Ki > 10000 nM T13644 CBV2X0 11963995 Ki > 10000 nM T13644 CW7I8U 13690207 Ki = 5.012 nM T13644 C8OU7I 15429504 IC50 = 5.6 nM T13644 CEO3F0 15585102 IC50 = 18.5 nM T13644 CC2YJ8 16062553 Ki > 10000 nM T13644 C3H1RT 16062555 Ki > 10000 nM T13644 C1LH5T 16062816 Ki > 10000 nM T13644 C1GKF8 16130982 Ki = 0.61 nM T13644 CW20OC 16144977 IC50 = 171 nM T13644 CS6A3Z 16145268 IC50 = 2276 nM T13644 CN3LS1 16145579 IC50 = 89.9 nM T13644 C72MUC 16146425 IC50 = 292 nM T13644 CD91IL 16148220 IC50 = 1127 nM T13644 C59OUC 16148481 Ki = 199.53 nM T13644 CJG1X9 16148596 Ki = 7.943 nM T13644 CNY09C 16148922 Ki = 1000 nM T13644 CP0DC8 16149640 Ki = 0.631 nM T13644 CDPC19 16149975 Ki = 1.585 nM T13644 C0SE6V 16150676 Ki = 0.631 nM T13644 CSP6A9 16150915 Ki = 0.631 nM T13644 C6N7SR 16151159 Ki = 25.12 nM T13644 C2B9IL 16151570 IC50 = 789 nM T13644 CQM8J1 16151781 IC50 = 210 nM T13644 CM8UF7 16151826 IC50 > 1000 nM T13644 CJ7UT6 16151923 IC50 = 325 nM T13644 CIM03U 16152257 IC50 = 135 nM T13644 CU7X6V 16153077 IC50 = 116 nM T13644 CK4O1V 16153193 IC50 = 263 nM T13644 C16LMW 16153418 IC50 = 980 nM T13644 CO0LG7 16154000 IC50 > 1000 nM T13644 CX4RM8 16154096 IC50 = 57 nM T13644 COYU86 16156815 Ki = 1000 nM T13644 CI3FW1 16157160 IC50 = 144 nM T13644 C7GN0S 16157479 Ki = 0.7943 nM T13644 CQL5O0 16181427 IC50 = 150 nM T13644 C2CUY9 16181428 IC50 > 1000 nM T13644 CUH8D7 16737812 IC50 > 1000 nM T13644 C8QIT3 16737813 IC50 > 1000 nM T13644 CNP36U 16737814 IC50 = 251 nM T13644 C7Q6JL 16738359 IC50 = 694 nM T13644 CJ9K1C 24740750 Ki > 10000 nM T13644 CS6VO9 24740751 Ki > 10000 nM T13644 CA4K0B 24740752 Ki > 10000 nM T13644 C4N3AX 24740753 Ki > 10000 nM T13644 COQU12 24740861 Ki > 10000 nM T13644 CAD4S1 24740862 Ki > 10000 nM T13644 C67YVI 24740863 Ki > 10000 nM T13644 CO0IF5 24740864 Ki > 10000 nM T13644 C6F1RZ 24777672 IC50 > 1000 nM T13644 C5GZO7 24858018 IC50 = 38 nM T13644 CV1U7H 24858920 IC50 = 4.5 nM T13644 C0UB7K 24859055 IC50 = 6.3 nM T13644 CQCW58 24859056 IC50 = 7.1 nM T13644 CT6J2A 24859195 IC50 = 19 nM T13644 CUDV69 24859196 IC50 = 12 nM T13644 C45NYA 24859341 IC50 = 15 nM T13644 C4AB6I 24859342 IC50 = 14 nM T13644 CH50QU 24859494 IC50 = 6 nM T13644 C8L2KJ 24859495 IC50 = 53 nM T13644 CDS6W5 24859645 IC50 = 20 nM T13644 CHF20D 24859646 IC50 = 36 nM T13644 CKH2R4 24859787 IC50 = 30 nM T13644 CT1BM6 24859788 IC50 = 28 nM T13644 C2IKX3 24859919 IC50 = 69 nM T13644 C5OQ2X 24859920 IC50 = 45 nM T13644 CSZ73L 24860057 IC50 = 50 nM T13644 C36ZHQ 24860058 IC50 = 31 nM T13644 CVL48C 24860201 IC50 = 19 nM T13644 C20ZFS 24860202 IC50 = 69 nM T13644 CHKC79 25187396 IC50 > 1000 nM T13644 C4YXJ1 25187398 IC50 = 153 nM T13644 CO9PI7 25187400 IC50 = 182 nM T13644 C8C9PL 25187679 IC50 = 162 nM T13644 C9ECD8 25187681 IC50 = 54 nM T13644 C43OES 25187683 IC50 > 500 nM T13644 CNTB73 25187685 IC50 = 119 nM T13644 C1IUQ2 25187953 IC50 = 316 nM T13644 CQ3F8L 25187955 IC50 = 9.1 nM T13644 CS2ZV1 25188218 IC50 = 403 nM T13644 CLI2U1 25188220 IC50 = 300 nM T13644 CNDU95 25188496 IC50 = 400 nM T13644 C7KF8N 25188776 IC50 = 910 nM T13644 CCHN50 25188780 IC50 = 515 nM T13644 C3T8DA 25189052 IC50 = 3.9 nM T13644 CI21ED 25189054 IC50 = 260 nM T13644 C97LHK 25189325 IC50 = 50 nM T13644 CEG4J0 25189327 IC50 = 105 nM T13644 CT5P4U 25204216 IC50 = 4 nM T13644 CSQH26 42637069 IC50 = 681 nM T13644 CJ1S9K 42637136 IC50 = 253 nM T13644 C3NYM8 42637137 IC50 > 1000 nM T13644 CJ47CL 42637210 IC50 > 1000 nM T13644 CR3A8Q 42637283 IC50 = 463 nM T13644 CENZ47 42637363 IC50 > 1000 nM T13644 CX0JC7 42637503 IC50 = 158 nM T13644 C90LHS 42637563 IC50 = 252 nM T13644 C80WBK 42637632 IC50 = 410 nM T13644 CR49YE 42637984 IC50 > 1000 nM T13644 CEFO24 42638065 IC50 = 60 nM T13644 CF5JK4 42638066 IC50 = 72 nM T13644 CHY04A 44290718 IC50 > 100 nM T13644 C16BKW 44290734 IC50 > 100 nM T13644 CW76YB 44290735 IC50 > 100 nM T13644 CA6IS7 44290766 IC50 = 15.6 nM T13644 C6BZ1J 44298104 Ki = 171 nM T13644 CCXL10 44298113 Ki = 51 nM T13644 CYW8O0 44298130 Ki = 108 nM T13644 CB9JK1 44298131 Ki = 53 nM T13644 CJ5WL8 44298155 Ki = 103 nM T13644 CHL57J 44298156 Ki = 379 nM T13644 CP61LB 44298165 Ki = 1560 nM T13644 CM0B6J 44298166 Ki = 1600 nM T13644 C8XZR7 44298169 Ki = 166 nM T13644 C0DPX7 44298171 Ki = 192 nM T13644 C62OEU 44298177 Ki = 495 nM T13644 CS9JW8 44298178 Ki = 838 nM T13644 C20MBI 44298179 Ki = 269 nM T13644 C3QBP0 44298188 Ki = 111 nM T13644 C1R3QD 44298189 Ki = 18 nM T13644 C5RJ7U 44298195 Ki = 120 nM T13644 C8N3EJ 44298197 Ki = 290 nM T13644 CZU05A 44298214 Ki = 1350 nM T13644 CQUS98 44298218 Ki = 382 nM T13644 COTK07 44298219 Ki = 385 nM T13644 CAJO07 44298231 Ki = 243 nM T13644 C9S4IX 44298232 Ki = 126 nM T13644 CB1A3K 44298235 Ki = 152 nM T13644 C2TQ1V 44298248 Ki = 124 nM T13644 C3WFV5 44298250 Ki = 57 nM T13644 CVW19Y 44298328 Ki = 93 nM T13644 CT94HY 44298329 Ki = 170 nM T13644 CL4F1V 44298378 Ki = 175 nM T13644 CMO1Q9 44298441 Ki = 38 nM T13644 C8Y9ZP 44298443 Ki = 85 nM T13644 CUSR45 44298468 Ki = 482 nM T13644 C8EN2H 44298469 Ki = 397 nM T13644 CWE7Q0 44298482 IC50 > 1000 nM T13644 CF69PL 44298522 Ki = 271 nM T13644 CRQJ98 44308836 Ki = 3614 nM T13644 CRFM02 44308969 Ki = 2950 nM T13644 C40MJU 44308970 Ki = 0.66 nM T13644 C9KR7Q 44309052 Ki = 3688 nM T13644 C4YG1S 44311590 IC50 = 345 nM T13644 CY0OV9 44311591 IC50 = 273 nM T13644 C29GQB 44311601 IC50 = 3.4 nM T13644 CC8DS0 44311602 IC50 > 1000 nM T13644 C5KST2 44311690 IC50 = 975 nM T13644 C6N4MH 44311691 IC50 > 10000 nM T13644 CIR4G6 44311695 IC50 > 1000 nM T13644 CTG6X5 44311696 IC50 = 618 nM T13644 C7Y8SF 44311697 IC50 > 1000 nM T13644 CK52MY 44311702 IC50 = 713 nM T13644 CX39CV 44311703 IC50 > 1000 nM T13644 C5RM2A 44311730 IC50 = 500 nM T13644 CBG70T 44311731 IC50 = 633 nM T13644 CQH20F 44311765 IC50 > 1000 nM T13644 CZG4K6 44311836 IC50 > 1000 nM T13644 CWNP79 44311837 IC50 = 290 nM T13644 CWSF38 44311868 IC50 > 1000 nM T13644 C2T0YP 44311869 IC50 = 280 nM T13644 C1ONB3 44311870 IC50 = 81 nM T13644 C1GY0F 44311912 IC50 > 1000 nM T13644 C14DIH 44311913 IC50 > 1000 nM T13644 C1X4TI 44311914 IC50 = 13.1 nM T13644 C64WAE 44311958 IC50 = 381 nM T13644 CFT90E 44311959 IC50 > 1000 nM T13644 C3PQD0 44311960 IC50 = 445 nM T13644 CS7PB4 44312258 IC50 > 10000 nM T13644 C5PE1D 44325273 IC50 = 1258 nM T13644 CN96LS 44332643 Ki = 84 nM T13644 C1P0QV 44332931 Ki = 1.7 nM T13644 CAG1Z4 44354386 Ki = 3750 nM T13644 C3QZH1 44354398 Ki = 5250 nM T13644 CHP41F 44363816 Ki = 1290 nM T13644 CH2DN4 44367916 IC50 > 1000 nM T13644 CM9YQ0 44367953 IC50 > 1000 nM T13644 C5W4YL 44368019 IC50 > 10000 nM T13644 CO6ZJ9 44368020 IC50 = 595 nM T13644 CQ5T1D 44368043 IC50 = 171 nM T13644 C1SWO5 44368044 IC50 = 697 nM T13644 C29EZK 44368080 IC50 = 9.7 nM T13644 C9ZW6U 44368093 IC50 = 325 nM T13644 C71URM 44368094 IC50 = 12 nM T13644 CC1ZP9 44368109 IC50 > 1000 nM T13644 CQ7OP1 44368112 IC50 = 186 nM T13644 C0EW4I 44368117 IC50 = 61 nM T13644 C6TNZ9 44368144 IC50 > 10000 nM T13644 C53IAG 44368153 IC50 = 14 nM T13644 CKU8J7 44368156 IC50 = 13 nM T13644 CR12GB 44368157 IC50 = 13 nM T13644 C50DMO 44368226 IC50 > 10000 nM T13644 CN31HS 44368398 IC50 = 319 nM T13644 C2RC0P 44368406 IC50 > 1000 nM T13644 CB1HC8 44368422 IC50 > 1000 nM T13644 C27DLY 44368489 IC50 > 1000 nM T13644 CWHK38 44377332 Ki > 10000 nM T13644 CVH1O7 44377366 Ki > 5000 nM T13644 CRC2N1 44377555 Ki = 1700 nM T13644 CS1WT5 44377591 Ki = 10000 nM T13644 C3LUY8 44377623 Ki = 8900 nM T13644 CQD0P4 44377645 Ki > 5000 nM T13644 CWNF42 44385504 Ki = 410 nM T13644 CAFD79 44385508 Ki = 400 nM T13644 CHY14B 44385591 Ki = 240 nM T13644 CJQI19 44385652 Ki = 250 nM T13644 CG12HD 44385712 Ki = 700 nM T13644 C8MU5C 44385757 Ki = 1400 nM T13644 C0LRT9 44386389 Ki = 500 nM T13644 C1EVK8 44387399 Ki = 802 nM T13644 C6U9VC 44388027 IC50 = 254 nM T13644 C2IW5J 44388028 IC50 > 1000 nM T13644 C27ANT 44388029 IC50 > 1000 nM T13644 CHQK20 44388035 IC50 > 1000 nM T13644 CI9XS1 44388036 IC50 > 1000 nM T13644 CD4BX6 44388037 IC50 > 1000 nM T13644 CDS08Z 44388038 IC50 > 1000 nM T13644 CZA03Y 44388040 IC50 > 1000 nM T13644 C21WBR 44388043 IC50 > 1000 nM T13644 C7VK6B 44388052 IC50 > 1000 nM T13644 CT93BI 44388060 IC50 > 1000 nM T13644 C4E5VS 44388061 IC50 > 1000 nM T13644 C7P5RO 44388066 IC50 > 1000 nM T13644 C7T8IY 44388069 IC50 > 1000 nM T13644 C2TWO3 44388070 IC50 > 1000 nM T13644 CDBE87 44388075 IC50 > 1000 nM T13644 C25GWK 44388078 IC50 > 1000 nM T13644 CT93LV 44388079 IC50 > 1000 nM T13644 CX54SC 44388083 IC50 > 1000 nM T13644 C2C0RU 44388084 IC50 = 620 nM T13644 C5SMA2 44388085 IC50 > 1000 nM T13644 C26OCG 44388086 IC50 > 1000 nM T13644 C8SR2O 44388087 IC50 > 1000 nM T13644 CHL5T1 44388088 IC50 > 1000 nM T13644 C4VNC2 44388089 IC50 > 1000 nM T13644 C1IH3T 44388090 IC50 > 1000 nM T13644 CNC91I 44388093 IC50 = 311 nM T13644 CN45OF 44388095 IC50 > 1000 nM T13644 C82HJL 44388104 IC50 > 1000 nM T13644 CV6T2H 44388105 IC50 > 1000 nM T13644 CLC0N2 44388106 IC50 > 1000 nM T13644 C0VO1K 44388107 IC50 > 1000 nM T13644 CM5O3B 44388108 IC50 > 1000 nM T13644 CAF02P 44388109 IC50 > 1000 nM T13644 C23XBM 44388110 IC50 = 772 nM T13644 CPX74G 44388112 IC50 > 1000 nM T13644 CG9SA3 44388114 IC50 > 1000 nM T13644 C2C4MH 44388116 IC50 > 1000 nM T13644 CW1EL5 44388118 IC50 > 1000 nM T13644 CN0K3V 44388119 IC50 > 1000 nM T13644 CE8DH4 44388120 IC50 > 1000 nM T13644 C1A0OY 44388121 IC50 > 1000 nM T13644 CS53NP 44388122 IC50 = 900 nM T13644 CX67WG 44388123 IC50 = 536 nM T13644 CB50EK 44388124 IC50 = 953 nM T13644 C9SN1X 44388132 IC50 > 1000 nM T13644 C6W4YT 44388133 IC50 > 1000 nM T13644 CMTN20 44388134 IC50 > 1000 nM T13644 CAK42W 44388135 IC50 > 1000 nM T13644 CTW48B 44388136 IC50 > 1000 nM T13644 C4P1AS 44388137 IC50 > 1000 nM T13644 CEAZ82 44388138 IC50 > 1000 nM T13644 C1KMT8 44397389 Ki = 100 nM T13644 CN6Z8C 44397648 Ki = 97 nM T13644 CRW0M6 44397706 Ki = 41 nM T13644 CM1R8X 44400000 IC50 = 389 nM T13644 CP89CS 44400135 IC50 > 1000 nM T13644 CV4PO0 44403186 IC50 > 1000 nM T13644 C8MEP3 44403194 IC50 > 1000 nM T13644 C9B3AP 44403195 IC50 > 1000 nM T13644 C29GND 44403204 IC50 > 1000 nM T13644 CM3KG6 44403206 IC50 > 1000 nM T13644 C0DG2C 44403217 IC50 > 1000 nM T13644 C9MBD4 44403227 IC50 > 1000 nM T13644 CLH53T 44403242 IC50 > 1000 nM T13644 CIEM04 44403248 IC50 > 1000 nM T13644 C1BY2P 44444935 IC50 > 1000 nM T13644 CH17TI 44560858 IC50 > 1000 nM T13644 C2AZY7 44560859 IC50 > 1000 nM T13644 C2I8NB 44560860 IC50 > 1000 nM T13644 C4XRT0 44560861 IC50 = 384 nM T13644 C21TZI 44560862 IC50 > 1000 nM T13644 C2YM5N 44560863 IC50 = 451 nM T13644 CS39FB 44560864 Ki = 93 nM T13644 CU3FD2 44560865 Ki = 50 nM T13644 C8IKU1 44560866 IC50 = 827 nM T13644 CTQ83Z 44560867 IC50 = 102 nM T13644 CQC29N 44560868 IC50 = 340 nM T13644 C47MDA 44560869 IC50 = 155 nM T13644 CHAJ41 44560870 IC50 = 54 nM T13644 CT0A9U 44560871 IC50 = 972 nM T13644 CM0T9R 44560872 IC50 = 124 nM T13644 CO2J6R 44560873 IC50 = 88 nM T13644 CKQD64 44560874 IC50 = 138 nM T13644 CEK26Y 44560875 IC50 = 255 nM T13644 CBL1P7 44560876 IC50 = 162 nM T13644 CY47DM 44560877 IC50 = 328 nM T13644 C5OZD1 44560878 IC50 = 336 nM T13644 CFT47C 44560898 IC50 = 661 nM T13644 CAO7R0 44560899 IC50 = 157 nM T13644 C80ZCF 44560900 IC50 = 120 nM T13644 CATH94 44560901 IC50 = 50 nM T13644 C2AXG6 44560902 IC50 = 90 nM T13644 COQ9W7 44560903 IC50 = 346 nM T13644 CLZ23V 44560904 IC50 > 1000 nM T13644 C0OKG2 44560905 IC50 = 8.3 nM T13644 CPIW17 44560906 IC50 > 1000 nM T13644 CFR3Y5 44560907 IC50 > 1000 nM T13644 CS85LR 44560908 IC50 > 1000 nM T13644 C6K1FI 44577218 IC50 > 1000 nM T13644 CAJ15T 44577219 IC50 = 452 nM T13644 CQD56E 44577220 IC50 = 112 nM T13644 CV18IC 44577221 IC50 = 359 nM T13644 CLJD09 45102042 IC50 = 1320 nM T13644 C63YJS 45139239 IC50 = 200 nM T13644 C63XPN 45267999 IC50 = 312 nM T13644 CF09UA 45268875 IC50 = 344 nM T13644 C2PNH4 45272264 IC50 > 1000 nM T13644 CFL9K7 45273129 IC50 = 112 nM T13644 C9Z4MR 45273130 IC50 = 234 nM T13644 C4RGN0 45273131 IC50 = 17 nM T13644 CCJ08W 46830055 IC50 = 24.2 nM T13644 CH18QA 46882131 Ki > 10000 nM T13644 CBZ3T9 46882132 Ki > 10000 nM T13644 C6KBJ2 46882133 Ki > 10000 nM T13644 CNL16U 46882180 Ki > 10000 nM T13644 CCX75M 46882181 Ki > 10000 nM T13644 C2BOJ6 46882182 Ki > 10000 nM T13644 C9ASC1 46882224 Ki > 10000 nM T13644 CB38SE 46882225 Ki > 10000 nM T13644 CP2N1U 46882226 Ki > 10000 nM T13644 CJ3Q6B 46882227 Ki > 10000 nM T13644 CRYQ47 46882445 Ki > 10000 nM T13644 CRZ1B0 46882446 Ki > 10000 nM T13644 CNEZ46 46882447 Ki > 10000 nM T13644 C8D1OR 46882448 Ki > 10000 nM T13644 CZ0G2R 46882449 Ki > 10000 nM T13644 CR37UF 46882513 Ki > 10000 nM T13644 CF3L8U 46882514 Ki > 10000 nM T13644 C91WKZ 46882515 Ki > 10000 nM T13644 CX21JH 46882516 Ki > 10000 nM T13644 CBJ92C 46882517 Ki > 10000 nM T13644 C8N3KX 46882577 Ki > 10000 nM T13644 CAH31I 46882578 Ki > 10000 nM T13644 CD2NL0 46882579 Ki > 10000 nM T13644 C9B0DF 46882620 Ki > 10000 nM T13644 CJ8I4L 46882621 Ki > 10000 nM T13644 C2YMA7 46882622 Ki > 10000 nM T13644 CD0VH7 46882664 Ki > 10000 nM T13644 C50YRJ 46882665 Ki > 10000 nM T13644 CXFV62 46882666 Ki > 10000 nM T13644 CR07WV 46882667 Ki > 10000 nM T13644 CF1HC7 46882668 Ki > 10000 nM T13644 CVIU56 46882708 Ki > 10000 nM T13644 C8S4LN 46882709 Ki > 10000 nM T13644 CJ7GM9 46882746 Ki > 10000 nM T13644 C6OM5H 46882789 Ki > 10000 nM T13644 C5MV8K 46882790 Ki > 10000 nM T13644 C6RD3V 46882791 Ki > 10000 nM T13644 C1WUF9 46882831 Ki > 10000 nM T13644 C5LM3W 46882832 Ki > 10000 nM T13644 CU1D6I 46902023 IC50 = 380 nM T13644 C84ZTC 49865341 IC50 > 1000 nM T13644 C3VZ4U 49865342 IC50 = 892 nM T13644 CGYR09 49865343 IC50 = 25 nM T13644 C35WID 49865344 IC50 > 1000 nM T13644 C0RK7G 49865345 IC50 = 1000 nM T13644 C4YLM7 49865346 IC50 > 1000 nM T13644 CZ4RI1 49865347 IC50 = 92.5 nM T13644 C9SNL1 52941607 IC50 = 8400 nM T13644 C40ZRY 52948630 IC50 = 500 nM T13644 CED3O6 53473658 IC50 = 13 nM T13644 CE7J0U 53473659 EC50 = 0.87 nM T13644 CY0G2K 53473744 EC50 = 0.35 nM T13644 CBQG96 53473824 EC50 = 0.23 nM T13644 CW53YV 53473917 IC50 = 131 nM T13644 C87SME 53474004 EC50 = 41 nM T13644 C7EO1Z 53474005 EC50 = 164 nM T13644 CY3M2A 53474090 EC50 = 299 nM T13644 C6EIJ5 54586681 Ki = 0.79 nM T13644 C9JHI4 56664813 Ki = 1.2 nM T13644 C8ZW3O 56927659 EC50 = 0.95 nM T13644 CHK8T1 56945132 Ki = 6628 nM T13644 C73XBL 57384077 IC50 = 11 nM T13644 C3KC9Z 57398462 IC50 = 3.5 nM T13644 C29YCJ 59411406 IC50 = 75.4 nM T13644 C97DHU 70682466 IC50 = 7 nM T13644 C4KWV3 70682467 IC50 = 16 nM T13644 CTVI05 70683416 IC50 = 329 nM T13644 C6CWV8 70684549 IC50 = 290 nM T13644 C9F5ZM 70684550 IC50 = 44 nM T13644 C1GN5V 70688791 IC50 = 10 nM T13644 CA7PZ9 70688792 IC50 = 21 nM T13644 C17MXW 70688793 IC50 = 180 nM T13644 CV42WQ 70689221 IC50 = 235 nM T13644 C3P0AN 70689413 IC50 = 205 nM T13644 CP58HL 70689414 IC50 = 98 nM T13644 CB14OW 70689415 IC50 = 172 nM T13644 CNZC97 70689723 IC50 = 112 nM T13644 CVSJ38 70690870 IC50 = 19 nM T13644 C2WQM9 70691295 IC50 > 1000 nM T13644 C5E8MY 70693613 IC50 = 175 nM T13644 C3TZ9U 70695246 IC50 = 273 nM T13644 C34XGS 70695722 IC50 = 82 nM T13644 CIPF50 70695723 IC50 = 308 nM T13644 CMS6J5 70697098 IC50 = 390 nM T13644 C84WJI 70697099 IC50 = 63 nM T13644 CPDJ19 71450468 IC50 = 2.3 nM T13644 CL01IH 71452297 IC50 = 58 nM T13644 C5ZKN6 71452298 IC50 = 0.76 nM T13644 CHQ1F0 71452299 IC50 = 2.8 nM T13644 CZI84F 71454093 IC50 = 1.1 nM T13644 C6PX9L 71457622 IC50 = 7.2 nM T13644 CF08XL 71458043 Ki = 1200 nM T13644 COJ85G 71459516 IC50 = 0.7 nM T13644 CU82HG 71460000 IC50 = 750 nM T13644 CETP14 71461260 IC50 = 0.97 nM T13644 CPC69G 71461645 Ki = 3100 nM T13644 CLAV92 71461684 IC50 > 1000 nM T13644 C1NZU3 71461685 IC50 > 1000 nM T13644 CH2CE8 71462982 IC50 = 19 nM T13644 C9R4EX 71462983 IC50 = 0.78 nM T13644 CQ4WG2 71462984 IC50 = 6.9 nM T13644 CFKH42 71717904 IC50 = 161 nM T13644 CGDO59 72947672 Ki = 4.24 nM T13644 CIO28F 73345407 Ki = 66 nM T13644 CMN6X8 73345525 IC50 = 403 nM T13644 C70XZC 73345528 IC50 = 3.1 nM T13644 CXGJ67 73345700 IC50 = 186 nM T13644 CV23JS 73345701 IC50 = 1000 nM T13644 C81UME 73345740 Ki = 709 nM T13644 CP6I2K 73346796 Ki = 11 nM T13644 CX5VM1 73346900 IC50 > 10000 nM T13644 CA3MU5 73346903 IC50 = 4.3 nM T13644 C62NFY 73346927 Ki = 68.7 nM T13644 CK64MX 73346930 Ki = 584 nM T13644 C15CAN 73346972 Ki = 253 nM T13644 CD09FU 73347225 Ki = 1190 nM T13644 CI4L6W 73347226 Ki = 568 nM T13644 CGM61R 73348311 IC50 = 0.84 nM T13644 CN1FD2 73348312 Ki = 0.9 nM T13644 C01GIQ 73348427 Ki = 576 nM T13644 C7Y9ZT 73348428 Ki = 23.6 nM T13644 CFLT50 73348719 IC50 > 100 nM T13644 C75NBQ 73348741 Ki = 371 nM T13644 C5MNX3 73348742 Ki = 210 nM T13644 CL94MY 73350006 Ki = 91.4 nM T13644 C0N6XK 73350010 Ki = 330 nM T13644 CTV30F 73350011 Ki = 390 nM T13644 CF2AK4 73350012 Ki = 537 nM T13644 C8N2HX 73351385 Ki = 5500 nM T13644 CK9CS4 73351516 Ki = 140 nM T13644 CNY13O 73351517 Ki = 148 nM T13644 CUN6L1 73351622 IC50 = 6.7 nM T13644 CC98JE 73351624 IC50 = 3.4 nM T13644 CWUH52 73351718 Ki = 40.2 nM T13644 CS9I4W 73351829 Ki = 231 nM T13644 CF70XH 73351873 IC50 > 1000 nM T13644 COID68 73352847 Ki = 28 nM T13644 CFB54J 73352985 Ki = 38.2 nM T13644 CKFV85 73353009 Ki = 797 nM T13644 CC45AV 73353272 IC50 = 187 nM T13644 C41OCY 73353278 IC50 > 100 nM T13644 CW54CU 73353340 IC50 > 1000 nM T13644 C2EWN7 73354353 Ki = 13 nM T13644 CWBQ47 73354354 Ki = 33 nM T13644 CK26MT 73354355 Ki = 200 nM T13644 CL7DT2 73354494 Ki = 1000 nM T13644 CA48EL 73354535 Ki = 425 nM T13644 CFK7Z3 73354633 IC50 = 664 nM T13644 C1UYL2 73354783 IC50 = 330 nM T13644 CG1CX0 73354798 IC50 > 100 nM T13644 CIVZ67 73354818 Ki = 100 nM T13644 CGCE64 73354819 Ki = 555 nM T13644 CC03JM 73355920 Ki = 11 nM T13644 CCV1Q6 73355921 Ki = 320 nM T13644 C1Y0CI 73356066 Ki = 1000 nM T13644 C52JAS 73356068 Ki = 315 nM T13644 CN5LG8 73356069 Ki = 450 nM T13644 C9GKV2 73356181 IC50 = 110 nM T13644 C7XFB6 73356331 IC50 = 40.7 nM T13644 CI02SE 73356366 Ki = 58 nM T13644 CW8L6C 76310862 IC50 > 1000 nM T13644 CHV6K7 76314485 IC50 = 98 nM T13644 C0PR3Y 76314486 IC50 > 1000 nM T13644 C94BWD 76314487 IC50 = 16 nM T13644 C25XKO 76314488 IC50 = 24 nM T13644 CS54IV 76321777 IC50 = 16 nM T13644 C94OAT 76321778 IC50 = 18 nM T13644 CU1IR8 76325402 IC50 = 2.4 nM T13644 CL09JQ 86279005 IC50 = 1.71 nM T13644 C3JOS4 86292350 Ki > 8597 nM T13644 CVLE34 86293506 Ki > 8580 nM T13644 C15VTO 86294248 Ki > 8615 nM T13644 CVIX61 90644974 Ki > 1109 nM T13644 C8T6AX 90644975 Ki = 1285 nM T13644 C3UK6H 90644976 Ki = 9 nM T13644 C9AF2G 90644977 Ki = 245 nM T13644 CB0G6C 90644978 Ki = 15.5 nM T13644 C3B7TY 90644979 EC50 = 348 nM T13644 CU73SD 90644980 Ki = 24 nM T13644 C2BAV8 90644981 EC50 = 2.88 nM T13644 CY1U7M 90644982 EC50 = 6.1 nM T13644 C8CH2G 90644983 Ki = 65 nM T13644 CVY1P0 90644984 EC50 = 21 nM T13644 CH70UW 90644985 EC50 = 13 nM T13644 C5C7KX 90644986 EC50 = 36 nM T13644 CJ1O0I 90644987 EC50 = 26 nM T13644 C14VQB 90644988 Ki > 12000 nM T13644 C5FA0O 90644989 EC50 = 59 nM T13644 CW49DL 90644990 EC50 = 11 nM T13644 CYZ3H7 90644991 Ki = 4.48 nM T13644 CFY3J1 90644992 EC50 = 0.516 nM T13644 CHM7U8 90644993 EC50 = 1.6 nM T13644 CN23IU 90644994 EC50 = 26 nM T13644 CC1F5D 90644995 EC50 = 22 nM T13644 CFZ30Q 90644996 Ki = 3.7 nM T13644 CL59GS 90644997 Ki = 30 nM T13644 C57FUD 90644998 Ki = 198 nM T13644 CS5GN4 90644999 Ki = 293 nM T13644 CX3DF2 90645000 Ki = 2336 nM T13644 CBLA30 90645001 Ki = 900 nM T13644 C6OG0I 90645002 Ki > 1200 nM T13644 CNMH13 90645003 Ki > 1128 nM T13644 CK3JP7 90645004 Ki > 1200 nM T13644 C96EKP 90645005 Ki = 5800 nM T13644 CSIB84 90645006 Ki > 1128 nM T13644 CGH28I 90645007 Ki = 17 nM T13644 C0ZQV6 90645008 Ki = 32 nM T13644 CSG76X 90645009 Ki > 12000 nM T13644 C7UNB3 90645010 Ki > 12000 nM T13644 CZU5O4 90645011 Ki = 97 nM T13644 CXOT87 90645012 Ki = 48 nM T13644 CX96KU 90645013 Ki = 4.15 nM T13644 C6G8DU 90645014 Ki = 236 nM T13644 CI58FM 90663867 IC50 = 357 nM T13644 CK62FO 90663868 IC50 = 243 nM T13644 C7AFD4 90663869 IC50 = 491 nM T13644 C94XTF 90663872 IC50 = 210 nM T13644 CA7W0U 90663873 IC50 = 757 nM T13644 C4EG8T 90663874 IC50 = 823 nM T13644 CW21UO 90663875 IC50 = 398 nM T13644 C7Q4PD 90665458 Ki = 17000 nM T13644 CR43ZL 90665459 Ki = 22000 nM T13644 CLK7C3 90665460 Ki = 2400 nM T13644 CZ0UC6 90665461 Ki = 4600 nM T13644 C0IBJ6 90665462 Ki = 3100 nM T13644 CPX0C9 90665463 Ki = 2700 nM T13644 C3UVC8 91936728 IC50 = 613 nM T13644 CT3UP7 91936729 IC50 > 1000 nM T13644 CD2E4L 101941290 IC50 = 404 nM T13644 C9KB3W 117711399 Ki > 8710 nM T13644 CFC1J5 118710523 IC50 = 1.97 nM T13644 C4X8NC 118710524 IC50 = 5.36 nM T13644 CK3WG9 118710525 IC50 = 0.64 nM T13644 C4NIK8 118710526 IC50 = 4.87 nM T13644 C3JAX9 118710527 IC50 = 0.15 nM T13644 CXV1C5 118710528 IC50 = 24 nM T13644 CA5TR0 118710529 IC50 = 1.72 nM T13644 CX9Q7Z 118710530 IC50 = 2.91 nM T13644 C27IPK 118710531 IC50 = 4.41 nM T13644 CGVS63 118710532 IC50 = 74.7 nM T13644 CVS94P 118710533 IC50 = 72.7 nM T13644 C9AZ1B 118710534 IC50 = 0.52 nM T13644 CR8X3P 118710535 IC50 = 6.12 nM T13644 C0YL9Z 118710536 IC50 = 2.4 nM T13644 CY26HQ 118710537 IC50 = 409 nM T13644 CTH52C 118718416 Ki = 2.512 nM T13644 CKQ4P6 118718462 IC50 = 539 nM T13644 C1Z7UJ 118718463 Ki = 199.53 nM T13644 CPYA80 118718465 IC50 = 821 nM T13644 CR61UD 118718466 IC50 = 525 nM T13644 CW64XN 118718500 IC50 = 1302 nM T13644 CB4D5T 118718501 IC50 = 177 nM T13644 CW5HG2 118718502 IC50 = 903 nM T13644 CC36KP 118718503 IC50 = 1196 nM T13644 C7FIQ1 118718504 IC50 = 435 nM T13644 CNBY57 118718505 IC50 = 1756 nM T13644 CPY4Q5 118718506 IC50 = 235 nM T13644 CO13JR 118718507 IC50 = 1228 nM T13644 CLFJ60 118718508 IC50 = 466 nM T13644 C13YUH 118718509 IC50 = 649 nM T13644 CP2O7U 118718510 IC50 = 619 nM T13644 CLDZ63 118718511 IC50 = 1609 nM T13644 CYQ7X2 118718854 IC50 = 136 nM T13644 CA6C4T 118719101 IC50 > 1000 nM T13644 CDZ3H4 118719196 IC50 = 326 nM T13644 CQRO32 118719197 IC50 = 381 nM T13644 CGXH91 118719198 IC50 = 197 nM T13644 C1QJX7 118719199 IC50 > 1000 nM T13644 C0GLC8 118719200 IC50 > 1000 nM T13644 C40NGQ 118719201 IC50 = 725 nM T13644 CK2W9T 118719202 IC50 = 447 nM T13644 CW4AT0 118719275 IC50 = 403 nM T13644 C5VWI1 118719303 IC50 = 1076 nM T13644 C5KGV7 122179447 IC50 = 15 nM T13644 CFO15B 122179448 IC50 = 538.6 nM T13644 CJP38S 122179449 IC50 = 25.3 nM T13644 C3FP8V 122179450 IC50 = 4.6 nM T13644 CQGW18 122179451 IC50 = 13.3 nM T13644 CYW75S 122179452 IC50 = 11.3 nM T13644 COHA53 122179453 IC50 = 20 nM T13644 CI8H9C 122179454 IC50 = 11.5 nM T13644 CKZ4X8 122179455 IC50 = 53.3 nM T13644 CZ6U4L 122179456 IC50 = 4.8 nM T13644 CS12JW 122179457 EC50 = 2.5 nM T13644 CEQ5M0 122179459 IC50 = 1.2 nM T13644 CNP81Q 122179460 IC50 = 1.2 nM T13644 C54KTN 122179461 IC50 = 0.4 nM T13644 C8DLB2 122179463 IC50 = 13.7 nM T13644 C56TKY 122179464 IC50 = 4.9 nM T13644 C49TGA 122179465 IC50 = 4.6 nM T13644 CWJ9C7 122179466 IC50 = 2.2 nM T13644 CI3L7J 122179467 IC50 = 3.5 nM T13644 C41LSM 122179468 IC50 = 3.3 nM T13644 C4U2EY 122179469 IC50 = 0.7 nM T13644 C24FUL 122179470 IC50 = 5.3 nM T13644 CN2FR7 122179471 IC50 = 2.2 nM T13644 CJ70OH 122179472 IC50 = 4.6 nM T13644 CBAO67 122179474 IC50 = 4.3 nM T13644 CQ0D2N 122179475 IC50 = 1.6 nM T13644 C7FA8O 122179476 IC50 = 2 nM T13644 CNGQ19 122179477 IC50 = 1.1 nM T13644 C9CLO5 122179478 IC50 = 0.4 nM T13644 CY6CB1 122179479 IC50 = 1 nM T13644 C4MZT8 122179480 IC50 = 1.4 nM T13644 CDQ37R 122179481 IC50 = 2.1 nM T13644 C6FME8 122179482 IC50 = 0.8 nM T13644 CO34VW 122179483 IC50 = 0.3 nM T13644 C34IFA 122186624 Ki = 180 nM T13644 CQ98SZ 122186625 Ki = 1500 nM T13644 CZB9X0 122186626 Ki = 51 nM T13644 CFDW42 122186627 Ki = 3.4 nM T13644 CAU9S5 122186628 Ki = 5.3 nM T13644 CG38WU 122186629 Ki = 60 nM T13644 CVF7Z5 122186630 Ki = 5.4 nM T13644 CGNZ17 122186631 Ki = 2 nM T13644 C3HMT2 122186632 Ki = 31 nM T13644 CK10DM 122186633 Ki = 26 nM T13644 CH1ZK4 122186634 Ki = 73 nM T13644 C5LZV2 122186635 EC50 = 20 nM T13644 CP70ZV 122186636 Ki = 24 nM T13644 CXMO69 122186637 Ki = 4.9 nM T13644 CROH96 122186638 EC50 = 61 nM T13644 CL8DW7 122186639 Ki = 37 nM T13644 CXJ64D 122186640 Ki = 1.3 nM T13644 CE7N5L 122186641 Ki = 510 nM T13644 CWY02F 122186642 Ki = 35 nM T13644 C78AGQ 122186643 EC50 = 1600 nM T13644 C98ULC 122186644 Ki = 32 nM T13644 C3A9YP 122186645 Ki = 32 nM T13644 CF7WO6 122186646 Ki = 330 nM T13644 CGJ8U0 122186647 Ki = 23 nM T13644 C1W9RN 122186648 Ki = 72 nM T13644 CWAP43 122186649 EC50 = 4200 nM T13644 CSV5L7 122186650 EC50 = 4800 nM T13644 CD2FQ6 122186651 Ki = 830 nM T13644 C63PDT 122186652 Ki = 160 nM T13644 C6XI1T 122186653 Ki = 1400 nM T13644 CUM1F8 122186654 Ki = 27 nM T13644 C62NBL 122186655 Ki = 1200 nM T13644 C0NCK8 122186656 Ki = 3400 nM T13644 CL37UN 122186657 EC50 = 4200 nM T13644 CL9IY6 127029888 IC50 = 391 nM T13644 C5RFV1 127029889 IC50 > 1333 nM T13644 CVQL89 127029890 EC50 > 1000 nM T13644 CZCQ82 127030226 EC50 = 1517 nM T13644 C7FD0M 127030227 EC50 = 26 nM T13644 C80JUT 127030228 EC50 = 181 nM T13644 C7YE3D 127030229 EC50 = 17 nM T13644 CF0S8I 127030230 EC50 = 6.4 nM T13644 CT9E3O 127030231 EC50 = 37 nM T13644 C48WEJ 127030232 IC50 = 225 nM T13644 CRV2K4 127030530 IC50 = 639 nM T13644 CJI5T4 127030531 IC50 = 43 nM T13644 C1F4OY 127030547 IC50 = 39 nM T13644 C3VFN1 127030548 EC50 = 199 nM T13644 C3TQ4U 127030549 EC50 = 0.46 nM T13644 C80CHF 127030550 IC50 = 2.6 nM T13644 CMKT63 127031154 EC50 = 88 nM T13644 CR87FU 127031155 IC50 = 18 nM T13644 CAV6G1 127031432 EC50 = 3.1 nM T13644 CMU7D8 127031454 EC50 = 50 nM T13644 CYKO59 127031455 IC50 = 141 nM T13644 C9FR7D 127031456 IC50 = 33 nM T13644 CY0EJ4 127031464 EC50 = 432 nM T13644 C4GH0Z 127031465 IC50 = 193 nM T13644 C1CR2M 127031771 EC50 = 4499 nM T13644 C2Z3TB 127031772 EC50 > 1000 nM T13644 C2GK1H 127031773 IC50 = 786 nM T13644 C89XCI 127031774 EC50 > 1000 nM T13644 CYAR63 127032340 IC50 = 230 nM T13644 C7XI2Z 127032341 EC50 = 1008 nM T13644 C1OE8W 127032342 IC50 = 25 nM T13644 C79DCQ 127032659 IC50 = 15 nM T13644 CDX69E 127032660 EC50 = 206 nM T13644 CMBA01 127032661 IC50 = 34 nM T13644 C2TH8G 127032662 IC50 = 10 nM T13644 C9DE0O 127032663 IC50 = 133 nM T13644 CJ1A5R 127033002 EC50 = 17 nM T13644 CLJ6G9 127033551 IC50 = 109 nM T13644 CE94YW 127033555 IC50 = 37 nM T13644 CPTV68 127033869 IC50 = 1333 nM T13644 C8QR3A 127033870 EC50 = 150 nM T13644 CU31BG 127033871 IC50 = 573 nM T13644 C8VP5X 127033872 EC50 = 938 nM T13644 CY81FE 127033873 EC50 = 405 nM T13644 CM7A1D 127033874 EC50 = 201 nM T13644 C5NU3M 127034125 EC50 = 17 nM T13644 C1FBI6 127034426 EC50 = 5.5 nM T13644 CLN17T 127034427 EC50 = 77 nM T13644 CMYQ47 127034428 EC50 = 7.4 nM T13644 CON9I2 127034429 EC50 = 4.8 nM T13644 CF27GZ 137062183 IC50 = 888.4 nM T13644 CE79SV 138377584 IC50 > 10000 nM T13644 C6ZU0A 145949555 IC50 > 20000 nM T13644 CE3D8P 145951877 IC50 > 20000 nM T13644 CI9BO4 145952624 IC50 > 20000 nM T13644 CL42TO 145953024 IC50 = 3120 nM T13644 CR2QH0 145957924 IC50 > 20000 nM T13644 CP25CA 145958767 IC50 = 6110 nM T13644 C01GKQ 145971455 IC50 > 20000 nM T13644 CG9KC4 145989896 IC50 = 119 nM T13644 CE76TG 42637005 IC50 = 701 nM T13644 C6ELN4 42637006 IC50 = 162 nM T13644 CS73LG 42637433 IC50 = 514 nM T13644 C6C3YF 45270549 IC50 = 618 nM T13644 C9Y3BS 45270550 IC50 > 1000 nM T13644 CQC51Z 45270552 IC50 > 1000 nM T13644 CXE30U 45271377 IC50 > 1000 nM T13644 D01BWV 9802572 Ki = 0.64 nM T13644 D01NID 44388055 IC50 > 1000 nM T13644 D02CQW 11847438 IC50 = 543 nM T13644 D02IXC 44403231 IC50 > 1000 nM T13644 D02NJV 44388048 IC50 = 789 nM T13644 D02OJQ 44388115 IC50 = 8 nM T13644 D02WOX 44388129 IC50 = 345 nM T13644 D03DRL 44388045 IC50 > 1000 nM T13644 D03SXC 44388041 IC50 > 1000 nM T13644 D03VHX 44388111 IC50 > 1000 nM T13644 D04EWA 44388034 IC50 > 1000 nM T13644 D04FPW 44388024 IC50 = 445 nM T13644 D04ORV 44388047 IC50 = 39 nM T13644 D04QBM 5311374 IC50 > 1000 nM T13644 D05COQ 11847588 IC50 = 38 nM T13644 D05XZA 44388071 IC50 > 1000 nM T13644 D06JWT 44388073 IC50 > 1000 nM T13644 D07DUF 44388130 IC50 > 1000 nM T13644 D07OSF 44388044 IC50 > 1000 nM T13644 D07WRP 15965425 Ki = 31 nM T13644 D09DAC 44388046 IC50 = 189 nM T13644 D09LHN 44311674 IC50 > 1000 nM T13644 D0A0DO 44388056 IC50 > 1000 nM T13644 D0A1XX 44388113 IC50 > 1000 nM T13644 D0BE3D 44388092 IC50 > 1000 nM T13644 D0C5RH 44388125 IC50 = 11 nM T13644 D0CC1P 44388042 IC50 > 1000 nM T13644 D0H0DC 44388051 IC50 = 905 nM T13644 D0H4WH 44388128 IC50 = 3.4 nM T13644 D0I9ME 44388074 IC50 > 1000 nM T13644 D0J5OY 44388022 IC50 = 222 nM T13644 D0M5LA 44388050 IC50 > 1000 nM T13644 D0N2MA 44388103 IC50 = 500 nM T13644 D0N4LH 44388065 IC50 > 1000 nM T13644 D0O4GU 44403230 Ki > 1000 nM T13644 D0P6ZZ 10581102 IC50 > 1000 nM T13644 D0R0OX 44388102 IC50 > 1000 nM T13644 D0R4IS 44388131 IC50 > 1000 nM T13644 D0S7YR 44388059 IC50 > 1000 nM T13644 D0T5RO 16129706 Ki = 0.1 nM T13644 D0W0AF 44388072 IC50 = 1029 nM T13644 D0WG0O 44388049 IC50 > 1000 nM T13644 D0Z0OF 44388094 IC50 = 617 nM T13644 D0Z1XY 44388064 IC50 > 1000 nM T13644 D0Z3LZ 44388023 IC50 = 52 nM T87024 D03SHD 892 IC50 = 100000 nM T87024 D04AIT 5280445 IC50 = 6400 nM T87024 D04NQI 2165 IC50 = 4000 nM T87024 D06DLI 4021 IC50 > 50000 nM T87024 D07HBX 338 Ki > 1800 nM T87024 D09CGE 24822371 Ki = 2.87 nM T87024 D09EGZ 2719 IC50 = 7000 nM T87024 D0A1PX 3394 IC50 = 305000 nM T87024 D0E6YQ 1935 IC50 = 12.21 nM T87024 D0K8KX 5280343 IC50 = 7940 nM T87024 D0N0ES 938 IC50 = 13100 nM T87024 D0W9LX 2585 IC50 = 30000 nM T87024 D03MFQ 9996409 IC50 = 14000 nM T87024 D05FGR 92337 IC50 = 280000 nM T87024 D07HZG 11516136 IC50 > 30000 nM T87024 D07SDQ 969516 IC50 = 3100 nM T87024 D09DLP 1646 IC50 = 100000 nM T87024 D09PYZ 44555286 IC50 = 10.5 nM T87024 D0U2BH 65064 IC50 = 500 nM T87024 D0U3EP 445154 IC50 = 1100 nM T87024 D03SLR 445858 IC50 > 100000 nM T87024 D0I3KT 44594137 IC50 = 1600 nM T87024 D0SF6C 10171904 EC50 = 69000 nM T87024 D03QTP 1697 Ki > 1000 nM T87024 D05UQD 656629 IC50 = 199.53 nM T87024 D06ABW 2788 IC50 = 100000 nM T87024 C0IN9E 11220755 Ki = 5 nM T87024 CJ8K9B 11674077 Ki = 5 nM T87024 C6QVA0 6508 IC50 > 100000 nM T87024 C82UCX 7087 Ki = 9.5 nM T87024 CG82OH 10390 Ki = 175 nM T87024 CCFH71 11313 Ki > 1000 nM T87024 C0VAW3 13735 IC50 < 3000 nM T87024 C6PUV9 16015 IC50 = 3000 nM T87024 CQ6L3K 16953 Ki = 890 nM T87024 CLV64D 16954 Ki = 116 nM T87024 CF3PD8 62344 IC50 = 600 nM T87024 CMVF62 66591 IC50 > 50000 nM T87024 CL0XM9 67232 IC50 > 50000 nM T87024 C39BCE 68275 IC50 < 3000 nM T87024 C7R6WV 82450 Ki = 64 nM T87024 C4HU6M 92095 IC50 > 100000 nM T87024 CSNZ31 95755 Ki = 4 nM T87024 C10EUP 97579 IC50 = 1000 nM T87024 CQ3LV1 124337 IC50 = 13400 nM T87024 CEXR79 160776 IC50 = 11200 nM T87024 CT5R3J 161557 IC50 = 12800 nM T87024 CPI83T 198909 IC50 = 11900 nM T87024 CZTD26 220436 IC50 = 1950 nM T87024 CD2NC9 234475 Ki = 37 nM T87024 CO03XS 260943 IC50 > 50000 nM T87024 CLG75C 384428 IC50 = 1200 nM T87024 CL8N5E 391870 Ki = 7 nM T87024 C28ACJ 396349 Ki = 26.2 nM T87024 CZ5S6D 459430 IC50 > 50000 nM T87024 CY5R1A 520360 EC50 = 4536000 nM T87024 C4V1HG 598987 IC50 = 900 nM T87024 CP58OT 637541 IC50 > 100000 nM T87024 CE1U8K 637829 EC50 = 20600 nM T87024 CZ0AH3 638278 IC50 = 19700 nM T87024 CC36US 689075 EC50 = 67700 nM T87024 CVUH50 701177 IC50 = 12000 nM T87024 CN1S9G 827500 Ki = 9 nM T87024 CT62ME 837893 Ki = 638 nM T87024 CO41FC 964143 Ki = 179.2 nM T87024 CX9LC5 1488786 Ki = 76 nM T87024 CXP17G 1604254 IC50 = 16700 nM T87024 CO1ZV8 2306524 Ki = 266.8 nM T87024 CKA4B8 2645568 IC50 = 10600 nM T87024 COY12A 2796853 IC50 = 23000 nM T87024 C6KGM2 2796861 IC50 = 13000 nM T87024 C0SJD8 2813371 IC50 = 700 nM T87024 C0SR3D 2819001 IC50 = 2300 nM T87024 C3LG9J 2826731 Ki = 0.8 nM T87024 CX2UN1 3589846 IC50 > 50000 nM T87024 CIK1P6 3620709 IC50 = 17600 nM T87024 CA1P8O 3743359 IC50 = 5000 nM T87024 CH9KY1 4127352 Ki = 4.31 nM T87024 C1HIJ5 5281292 IC50 = 2700 nM T87024 C20DJG 5281610 IC50 = 55400 nM T87024 CGS9B0 5281780 IC50 = 4700 nM T87024 CY28LS 5293755 Ki = 155.1 nM T87024 C6W1VC 5316144 IC50 > 50000 nM T87024 COA8T2 5316145 IC50 > 50000 nM T87024 CWQ8H9 5316884 IC50 = 17300 nM T87024 CF1V3Z 5318537 IC50 > 50000 nM T87024 CV3H5D 5319235 EC50 = 251500 nM T87024 CW1UM5 5357488 IC50 = 8400 nM T87024 C2SE9J 5369459 EC50 = 1040000 nM T87024 CN69HE 5375988 Ki = 95 nM T87024 CM7Z4V 5378081 Ki = 2.3 nM T87024 C1FAO0 5463186 Ki = 22 nM T87024 C0KSG2 5494423 IC50 = 180 nM T87024 C5ZS3K 5713403 Ki = 439.2 nM T87024 CV65ES 5919800 IC50 = 9700 nM T87024 CZ9Q1O 5928757 Ki = 325.2 nM T87024 CS80AZ 6435245 IC50 > 100000 nM T87024 CM56IW 6440783 IC50 = 300 nM T87024 CQ3S8L 6450842 Ki = 91.6 nM T87024 C45QJF 6474309 IC50 = 100 nM T87024 CSA24L 6474310 IC50 = 16400 nM T87024 CO5YF2 6476139 IC50 > 100000 nM T87024 CXE9B1 6506968 IC50 = 5700 nM T87024 C0QTS5 6518166 Ki = 13.65 nM T87024 C36LJK 9604154 Ki = 514.65 nM T87024 C56ITM 9835167 Ki = 4.9 nM T87024 C7ZM5D 9837643 Ki = 1.28 nM T87024 CWPO30 9839907 Ki = 5.9 nM T87024 C17JYE 9849211 IC50 = 15 nM T87024 CYLG46 9959612 IC50 = 8400 nM T87024 CS9VZ6 9972775 IC50 = 129000 nM T87024 CISM03 9976141 IC50 = 33600 nM T87024 CSZT84 9985405 IC50 = 32800 nM T87024 C2H0DW 9991705 EC50 = 12000 nM T87024 C7BLD1 10039500 IC50 = 5000 nM T87024 CSK82J 10042056 IC50 = 21000 nM T87024 CGO1C4 10051410 IC50 = 3100 nM T87024 CU5AE1 10064445 Ki = 19.97 nM T87024 CVK3F1 10066999 IC50 = 1600 nM T87024 CQ3WS6 10082261 EC50 = 24700 nM T87024 CZN01G 10107393 Ki = 0.74 nM T87024 CM0UC5 10125236 IC50 > 50000 nM T87024 C8R9HM 10133297 Ki = 1.29 nM T87024 CVX4J2 10143259 IC50 = 73 nM T87024 CTR45Y 10172574 IC50 = 4900 nM T87024 COH1K8 10184360 Ki = 0.11 nM T87024 C3EH5J 10220170 Ki = 3.04 nM T87024 COA56B 10236080 IC50 > 50000 nM T87024 CLV83M 10246831 Ki > 1000 nM T87024 CVO9F8 10308838 IC50 = 87800 nM T87024 C7FUL5 10311969 IC50 = 16 nM T87024 CN65TI 10315170 IC50 = 4500 nM T87024 C85AHL 10335228 Ki = 7.2 nM T87024 CN2ZH1 10364928 IC50 = 17700 nM T87024 CQ78FV 10392851 IC50 = 21300 nM T87024 CUY39V 10422457 Ki = 10 nM T87024 CT96UL 10426074 Ki = 1.7 nM T87024 CC9DU4 10444413 Ki = 46 nM T87024 CK09VZ 10471478 IC50 = 22000 nM T87024 CW0H6K 10496851 Ki = 0.8 nM T87024 CC78NM 10529819 EC50 = 112600 nM T87024 C75LHR 10547782 Ki = 0.9 nM T87024 CH2FE7 10637399 Ki > 4000 nM T87024 CYC50J 10745352 Ki = 0.17 nM T87024 CYF69B 10762840 Ki = 1.6 nM T87024 CDR68M 10815986 IC50 = 8000 nM T87024 CY3ED1 10844298 Ki = 5.4 nM T87024 CY5W6A 10889525 Ki > 1000 nM T87024 CFVS96 10895598 IC50 > 20000 nM T87024 C0WLA5 10914234 Ki = 32 nM T87024 C9ND4U 10922978 Ki = 64 nM T87024 CB6WU4 10936986 Ki = 2 nM T87024 CF6G9N 10947017 Ki = 339 nM T87024 C5L6OB 10956585 Ki = 4.4 nM T87024 CBP5V6 10978824 Ki = 11 nM T87024 CCH3F0 10983792 Ki > 2000 nM T87024 CS6UT3 11013106 Ki = 22 nM T87024 C8BW3U 11027604 IC50 = 1700 nM T87024 CNF04A 11054105 Ki = 242 nM T87024 CXQ7I8 11089783 Ki > 2000 nM T87024 C7WE6M 11103936 IC50 > 50000 nM T87024 CL2MI5 11110864 Ki = 4.5 nM T87024 CKMR07 11129817 Ki = 1.9 nM T87024 CILM15 11134806 IC50 = 2000 nM T87024 C35LNF 11139152 Ki > 2000 nM T87024 C9HEN8 11142607 Ki = 7.7 nM T87024 C9LVZ8 11351105 EC50 = 530 nM T87024 C0B6CE 11354073 IC50 = 0.3 nM T87024 CX1ND6 11455014 IC50 = 2425 nM T87024 C1DV2Z 11461081 IC50 > 100000 nM T87024 C8WI9Y 11488357 EC50 = 100 nM T87024 CH36VW 11500527 Ki = 12 nM T87024 CO97LY 11501341 Ki = 2.2 nM T87024 C4OS0M 11504350 EC50 = 13600 nM T87024 C91PCX 11507713 Ki = 15 nM T87024 C24RLF 11508700 IC50 = 81000 nM T87024 CK35JZ 11512035 IC50 = 6000 nM T87024 CK70GR 11512869 IC50 = 9900 nM T87024 COTH53 11516139 IC50 = 46000 nM T87024 CVPX30 11523521 IC50 = 57900 nM T87024 C58LDV 11529378 IC50 = 210000 nM T87024 CDT83G 11530779 IC50 = 20000 nM T87024 CBP8Y9 11532527 EC50 = 9200 nM T87024 C2IL9N 11543843 EC50 = 16000 nM T87024 CHF92A 11544421 Ki = 38 nM T87024 C4IP5W 11546946 EC50 = 8600 nM T87024 CHT39Z 11549051 IC50 > 6700 nM T87024 C8CA9X 11561538 EC50 = 2200 nM T87024 CM76TJ 11565846 IC50 = 12000 nM T87024 C2B6HV 11565868 IC50 = 77000 nM T87024 CKVN61 11566215 IC50 = 114000 nM T87024 COP47N 11573395 EC50 = 15400 nM T87024 CFP69L 11573705 IC50 = 41000 nM T87024 C5RNW0 11574638 EC50 = 16000 nM T87024 CS2WU3 11576068 EC50 = 4800 nM T87024 CJ73ZH 11580454 IC50 = 75000 nM T87024 C3YXZ7 11582291 IC50 = 11000 nM T87024 CF40ZR 11595039 Ki = 391 nM T87024 C1A7SE 11596660 EC50 = 4800 nM T87024 CR37EA 11602469 IC50 = 35000 nM T87024 C7ENB2 11609939 IC50 = 31600 nM T87024 CMQ38D 11619220 EC50 = 2100 nM T87024 CLI21W 11621627 IC50 = 5.2 nM T87024 CZ8E2P 11623805 Ki = 3.9 nM T87024 CO4Z7H 11626862 Ki = 80 nM T87024 CFXW58 11631766 Ki = 694.7 nM T87024 CWD47I 11638208 Ki = 32.5 nM T87024 CBI2Q1 11642048 EC50 = 440 nM T87024 C4A5YO 11644770 IC50 = 67000 nM T87024 CS48EP 11645550 IC50 = 70600 nM T87024 CR16HF 11649408 IC50 > 20000 nM T87024 C7FL0K 11657376 IC50 = 740 nM T87024 C9XE7B 11660650 Ki = 59 nM T87024 CGY2S9 11673829 IC50 = 83000 nM T87024 CLY02G 11682722 IC50 = 4200 nM T87024 C4G6YQ 11684817 EC50 = 3200 nM T87024 C2IW8S 11705141 EC50 = 13300 nM T87024 C73UBS 11709395 IC50 = 96300 nM T87024 C7ZRM9 11719190 EC50 = 5200 nM T87024 C2BDF9 11730513 IC50 = 1500 nM T87024 CD6S0B 11757331 IC50 > 50000 nM T87024 C0NC8U 11785317 IC50 = 57 nM T87024 C2LQ8I 11821524 Ki = 8.6 nM T87024 CQ26XH 11851431 IC50 = 2.4 nM T87024 CDB2Y5 11962185 IC50 = 15 nM T87024 CJD8H4 11964482 Ki = 10 nM T87024 C72CNY 12034742 EC50 = 10400 nM T87024 CDX43C 12179987 Ki = 2.2 nM T87024 CTWB58 13565967 EC50 = 2820 nM T87024 CO7QU8 13640229 Ki = 4.38 nM T87024 C1Y5TZ 13640230 Ki = 10.82 nM T87024 CM8N3F 13888657 IC50 = 13000 nM T87024 CDY85L 13888659 IC50 = 45600 nM T87024 CLV24A 14214498 IC50 = 2200 nM T87024 CQDV96 14804615 IC50 = 7800 nM T87024 CGC1O3 14818641 EC50 = 7950 nM T87024 C62KEJ 14837578 IC50 = 1900 nM T87024 C6JIA9 14977359 IC50 = 9000 nM T87024 CV3XL7 15086370 EC50 = 2580 nM T87024 CNC16Y 15086371 EC50 = 9520 nM T87024 CC4DY8 15228041 IC50 = 72900 nM T87024 CUO6L0 15521135 Ki = 0.13 nM T87024 CO37RN 15521136 Ki = 0.19 nM T87024 CULQ06 15521137 Ki = 0.27 nM T87024 CXD53V 15825666 IC50 > 100000 nM T87024 CD3KH2 15950376 Ki = 0.7 nM T87024 CN9U3G 16049314 Ki = 24.2 nM T87024 C4DO8C 16050931 EC50 = 810 nM T87024 C0Q2MC 16051586 EC50 = 180 nM T87024 CJOB87 16087291 Ki = 839.2 nM T87024 C78MGR 16087303 Ki = 232.7 nM T87024 C76FAU 16221445 Ki = 4.5 nM T87024 C5H6UD 16221447 Ki = 14.2 nM T87024 CR9F8B 16221507 Ki = 7.5 nM T87024 CQ62AD 16221508 Ki = 9 nM T87024 C3PW6R 16221509 Ki = 21 nM T87024 C9YTA6 16221511 Ki = 3.6 nM T87024 C0P3IZ 16221562 Ki = 5 nM T87024 CA4G1R 16221566 Ki = 8.5 nM T87024 CS0UT6 16221567 Ki = 15.5 nM T87024 C9JL5H 16221621 Ki = 6.8 nM T87024 C3TA8Q 16221676 Ki = 7.5 nM T87024 COA3D0 16659245 Ki = 1.5 nM T87024 CB7CP0 16659246 Ki = 12 nM T87024 C9N7PD 16659247 Ki = 1.2 nM T87024 CF4S8P 16659248 Ki = 5 nM T87024 CN5JH0 16659288 Ki = 67.58 nM T87024 CL84UE 16659290 Ki = 4.5 nM T87024 CDW95O 16659294 Ki = 3.8 nM T87024 CX4U1E 16659341 Ki = 16.5 nM T87024 C9F5PV 16659342 Ki = 2.9 nM T87024 C74ISD 16659343 Ki = 21.5 nM T87024 CDF25A 16659381 Ki = 2.9 nM T87024 CGI56O 16659384 Ki = 3.1 nM T87024 CX7LR3 16659421 Ki = 1.9 nM T87024 C2YE4L 16659422 Ki = 3.4 nM T87024 C0D7UN 16663275 Ki = 1.7 nM T87024 CLM19J 16664222 IC50 = 500 nM T87024 COS4Z8 16733863 Ki = 4.1 nM T87024 CVL3S7 16734166 Ki = 22.5 nM T87024 C0KTQ8 16753967 IC50 = 10200 nM T87024 CWUZ06 17758933 Ki = 13 nM T87024 CRS05M 17758934 Ki = 7.6 nM T87024 CC3O7A 17759055 Ki = 8.3 nM T87024 CPQ57L 17759056 Ki = 183 nM T87024 CV09PD 17759057 Ki > 1000 nM T87024 CLI57M 17759058 Ki = 7.4 nM T87024 C0A3SL 17759059 Ki = 658 nM T87024 CFE57D 17759060 Ki = 8.3 nM T87024 C9Q7KD 17759061 Ki = 147 nM T87024 CT58FH 17759200 Ki = 177 nM T87024 C5QKS4 17759203 Ki = 24.2 nM T87024 CH8P1M 17759204 Ki = 8.2 nM T87024 CIXG80 17759205 Ki = 38.5 nM T87024 CM4TX7 17759327 Ki > 180 nM T87024 CB63VN 17759328 Ki > 1000 nM T87024 CVG29B 17759329 Ki > 1000 nM T87024 CM4TH3 17759330 Ki > 1000 nM T87024 C8JL6K 17759331 Ki = 88 nM T87024 C8HFZ0 18149922 Ki = 103.62 nM T87024 C0ERF7 18149923 Ki = 107.6 nM T87024 C06QXP 18149927 Ki = 54.22 nM T87024 C1D4QK 18149928 Ki = 9.98 nM T87024 CRA2N7 18149931 Ki = 73.46 nM T87024 C5DFW9 18281386 Ki = 143.81 nM T87024 C3DE5H 19106793 Ki = 107.1 nM T87024 CZ6C2O 21176359 Ki = 106.46 nM T87024 C8T3HM 21299300 Ki = 1.1 nM T87024 CK54BE 21716170 EC50 = 5130 nM T87024 CWUS28 22361008 IC50 = 4600 nM T87024 C5ZOX7 22380809 Ki > 2000 nM T87024 C9N2FR 22692669 IC50 = 13000 nM T87024 C21BZS 23628239 Ki = 9.2 nM T87024 CG61EZ 23765385 IC50 = 7000 nM T87024 C6FM9C 24180452 IC50 = 6.9 nM T87024 CZGD65 24241910 Ki = 432.03 nM T87024 CCO5Y9 24742039 Ki = 7.93 nM T87024 C43RWH 24752854 IC50 = 100 nM T87024 C8JRW6 24754917 Ki = 377 nM T87024 CETG93 24754918 Ki = 205 nM T87024 CMT0Y8 24754920 Ki = 80 nM T87024 C3I5SN 24757878 IC50 = 81 nM T87024 CJFT24 24780524 IC50 = 185 nM T87024 C96MCU 24780657 IC50 = 137 nM T87024 C45EAK 24780800 IC50 = 35 nM T87024 C3C4NM 24780958 IC50 = 158 nM T87024 CH9E0S 24782384 IC50 = 1800 nM T87024 CYD31F 24782385 IC50 = 20000 nM T87024 C7L6CH 24782386 IC50 > 20000 nM T87024 CALC96 24782387 IC50 > 20000 nM T87024 CZBH76 24782389 IC50 = 600 nM T87024 CMV82Q 24785163 IC50 = 600 nM T87024 C72YPZ 24785412 IC50 = 1100 nM T87024 C26HTP 24785414 IC50 = 900 nM T87024 CIH92R 24785416 IC50 = 700 nM T87024 CNM5R6 24785417 IC50 = 900 nM T87024 C4TUW5 24785683 IC50 = 800 nM T87024 CIQ0M4 24785684 IC50 = 900 nM T87024 C18DSF 24785686 IC50 = 1100 nM T87024 CPHE83 24785954 IC50 = 600 nM T87024 CCG25U 24785955 IC50 = 1000 nM T87024 CKX8E0 24786215 IC50 = 700 nM T87024 C2YRX8 24786216 IC50 = 1300 nM T87024 C3T5DS 24786217 IC50 = 300 nM T87024 C63TMV 24786218 IC50 = 1100 nM T87024 CFW1V3 24786219 IC50 = 2700 nM T87024 CW37TI 24786220 IC50 > 20000 nM T87024 C7JPS0 24803728 IC50 = 74 nM T87024 CB4P9M 24804066 IC50 = 41 nM T87024 C8EY6Q 24804068 IC50 = 267 nM T87024 CPF80R 24804394 IC50 = 85 nM T87024 CWHM14 24814778 IC50 = 10000 nM T87024 COK6Y3 24822879 Ki = 1.5 nM T87024 CCL0P8 24858429 Ki = 152 nM T87024 CW8NE4 24896605 IC50 = 24 nM T87024 CYDL23 24952085 IC50 = 420 nM T87024 CD79SW 24954231 IC50 = 40500 nM T87024 CM7V5O 24954590 IC50 = 7500 nM T87024 CP5A0Z 24954962 IC50 = 29000 nM T87024 C1RB4M 24966387 IC50 = 3700 nM T87024 CHL57E 25014934 IC50 = 35 nM T87024 C75PBE 25015016 IC50 = 30 nM T87024 CCXN63 25110762 IC50 = 70 nM T87024 CH47IA 25110763 IC50 = 80 nM T87024 CHN93D 25145301 IC50 = 5000 nM T87024 CU45TK 25149265 IC50 = 9690 nM T87024 C3TF1N 25153233 IC50 = 270 nM T87024 C50PUD 25233595 Ki = 776 nM T87024 CR94SX 25233596 Ki = 5.7 nM T87024 C40XVQ 25233597 Ki > 4000 nM T87024 C3CLW6 25263467 EC50 = 12200 nM T87024 COWL38 25663159 Ki = 103.35 nM T87024 C8PKX4 31247355 Ki = 39.19 nM T87024 CU6X5C 42603587 Ki = 18.8 nM T87024 C0W5DV 42603588 Ki = 11.2 nM T87024 C9BH2X 42603729 Ki = 11.5 nM T87024 CZ1SP0 44124011 Ki = 22 nM T87024 CIYH27 44258702 IC50 = 5400 nM T87024 C8EV4N 44310689 Ki = 31 nM T87024 C8G7PI 44311003 Ki = 41 nM T87024 C9H4CZ 44313381 IC50 = 2700 nM T87024 CJ8SO9 44313401 IC50 = 1800 nM T87024 C9AT1P 44313410 IC50 = 10000 nM T87024 CS9A4Y 44313421 IC50 = 11000 nM T87024 C2KR9L 44391426 EC50 = 50600 nM T87024 CER5L0 44391470 EC50 = 2700 nM T87024 C1UZX2 44391471 EC50 = 62700 nM T87024 C2O6MY 44391488 EC50 = 48600 nM T87024 CHJG31 44391494 EC50 = 24500 nM T87024 C9NM2X 44391570 EC50 = 97000 nM T87024 CD9TR7 44403923 Ki = 150 nM T87024 C3AQE6 44408778 Ki > 1000 nM T87024 CAI52R 44408841 Ki = 500 nM T87024 C59USF 44408847 Ki = 7.5 nM T87024 C9SCY1 44408848 Ki = 21.5 nM T87024 CP7T2S 44410472 IC50 = 30 nM T87024 C2MT5J 44410474 IC50 = 74 nM T87024 CNJS75 44410489 IC50 = 5000 nM T87024 C5BK4F 44410504 IC50 = 152 nM T87024 CI5C0J 44410506 IC50 = 17 nM T87024 COA03X 44410508 IC50 = 3000 nM T87024 C3A9JI 44410509 IC50 = 6000 nM T87024 C0HG3W 44410511 IC50 = 160 nM T87024 CI0YG5 44410625 IC50 = 29 nM T87024 C76IRU 44410629 IC50 = 17 nM T87024 C8XPQ7 44410645 IC50 = 3000 nM T87024 CU5R6Z 44410681 IC50 = 6800 nM T87024 CU7K1S 44410738 IC50 = 54 nM T87024 CB5TU1 44411893 Ki = 177 nM T87024 C5P8QY 44411897 Ki = 48.3 nM T87024 CC73RW 44422929 Ki = 106 nM T87024 CRTD20 44422933 Ki = 2.9 nM T87024 C1QJY6 44425691 IC50 = 530 nM T87024 CI3A5Y 44425692 IC50 = 220 nM T87024 CCM4B6 44425693 IC50 = 280 nM T87024 C37DQY 44425694 IC50 = 86 nM T87024 CS1AP2 44425695 IC50 = 1900 nM T87024 C7F8GK 44425696 IC50 = 780 nM T87024 C30BMF 44425697 IC50 = 880 nM T87024 C0GD7L 44425707 IC50 = 680 nM T87024 C4SGC0 44425709 IC50 = 1000 nM T87024 C6YX3K 44425710 IC50 = 180 nM T87024 C4P6AD 44425712 IC50 = 900 nM T87024 CPJ0K2 44425713 IC50 = 190 nM T87024 CTOA30 44425715 IC50 = 360 nM T87024 CA1XZ5 44425716 IC50 = 60 nM T87024 CJV93D 44425718 IC50 = 600 nM T87024 CZH24M 44425720 IC50 = 650 nM T87024 C5T1KQ 44425721 IC50 = 450 nM T87024 CHD74S 44425722 IC50 = 540 nM T87024 C3O6AI 44425723 IC50 = 120 nM T87024 CXQ93D 44425724 IC50 = 140 nM T87024 CY65TM 44425725 IC50 = 180 nM T87024 C1F4JP 44427526 Ki = 1840 nM T87024 CX1VB2 44427527 Ki = 645 nM T87024 C8B2IN 44427528 Ki = 88 nM T87024 CSW0A7 44427529 Ki > 1000 nM T87024 C63DZH 44427530 Ki > 1000 nM T87024 C7P8IM 44428892 Ki = 25 nM T87024 C7J6ER 44428894 Ki = 34 nM T87024 CL3JI4 44428896 Ki = 36 nM T87024 C9RPI1 44428897 Ki = 25 nM T87024 CIM3V0 44428900 Ki = 6.8 nM T87024 CQ4TS5 44428902 Ki = 27 nM T87024 CD8LG5 44428903 Ki = 23 nM T87024 CAI1O7 44428904 Ki = 21 nM T87024 CV4Y7T 44432253 Ki = 16.8 nM T87024 C84YVS 44432254 Ki = 11.2 nM T87024 C6D9AI 44432255 Ki = 6.7 nM T87024 C7Y4RV 44432256 Ki = 13.1 nM T87024 C69JNA 44432257 Ki = 1.6 nM T87024 C5C2JX 44432258 Ki = 12.5 nM T87024 C0V9XC 44432259 Ki = 6.2 nM T87024 C2BOM0 44435362 IC50 = 2.8 nM T87024 C9CDJ4 44435363 IC50 = 2.5 nM T87024 CDKT27 44435364 IC50 = 3.5 nM T87024 CKB47T 44435365 IC50 = 3.5 nM T87024 C4Q2MH 44435366 IC50 = 27 nM T87024 CX51JK 44435367 IC50 = 12 nM T87024 C5B2KT 44435368 IC50 = 14 nM T87024 C4DF9U 44435369 IC50 = 17 nM T87024 CU85IX 44435370 IC50 = 46 nM T87024 C1RVA7 44435371 IC50 = 47 nM T87024 C35EIX 44435372 IC50 = 56 nM T87024 C1MXF7 44435378 IC50 = 3.2 nM T87024 CF3G6O 44435379 IC50 = 28 nM T87024 C31FSA 44435380 IC50 = 9 nM T87024 CK68EU 44435381 IC50 = 10 nM T87024 C9FPT6 44435382 IC50 = 12 nM T87024 C6TKA2 44435383 IC50 = 15 nM T87024 C2DXN4 44435384 IC50 = 3.5 nM T87024 C90BHK 44435385 IC50 = 25 nM T87024 C0F1LD 44435386 IC50 = 25 nM T87024 CK1LW9 44435387 IC50 = 16 nM T87024 CT3GE0 44435388 IC50 = 9.6 nM T87024 CQ9B8J 44435389 IC50 = 27 nM T87024 CR4K8U 44435390 IC50 = 45 nM T87024 CP78NT 44435391 IC50 = 81 nM T87024 C3JTA5 44435392 IC50 = 29 nM T87024 CJDU30 44435393 IC50 = 32 nM T87024 C1SCL8 44435394 IC50 = 39 nM T87024 C5TNV9 44435395 IC50 = 104 nM T87024 C1WIX8 44537956 IC50 = 2750 nM T87024 C0V7DG 44545776 IC50 = 23.1 nM T87024 C0Y2JB 44548006 IC50 = 470 nM T87024 CKV63Y 44548007 IC50 = 130 nM T87024 CC5LK7 44548162 IC50 = 200 nM T87024 C4ZF2H 44548163 IC50 = 1980 nM T87024 CBK2W7 44548164 IC50 = 170 nM T87024 CN3HV6 44548165 IC50 = 160 nM T87024 CZ03KC 44548166 IC50 = 3440 nM T87024 CO5FE2 44548167 IC50 = 3210 nM T87024 CFOB16 44548168 IC50 = 2190 nM T87024 CP9F4O 44548169 IC50 = 3620 nM T87024 CO19TF 44548342 IC50 = 2300 nM T87024 CHE3K1 44548343 IC50 = 810 nM T87024 C2XZ3E 44548344 IC50 = 1340 nM T87024 CK9W5J 44548345 IC50 = 2800 nM T87024 CDG2Q1 44548346 IC50 = 820 nM T87024 CZ4HL9 44548348 IC50 = 2950 nM T87024 C2LG9W 44548350 IC50 = 2160 nM T87024 CT9E6K 44548351 IC50 = 5440 nM T87024 C5G0JO 44548514 IC50 = 800 nM T87024 C48YRH 44548515 IC50 = 160 nM T87024 CM9BQ3 44548516 IC50 = 530 nM T87024 CI0HY6 44550347 Ki = 3.8 nM T87024 C27LAB 44552725 IC50 = 30.2 nM T87024 C5WQD8 44552727 IC50 = 47 nM T87024 C5LEV4 44554966 IC50 = 8 nM T87024 C3AU6G 44554967 IC50 = 35.8 nM T87024 CQL2Z1 44555120 IC50 = 4 nM T87024 CC9NG2 44555125 IC50 = 13.8 nM T87024 C4FW3G 44555283 IC50 = 25.7 nM T87024 CD3WK2 44555284 IC50 = 41.8 nM T87024 CXZS18 44555289 IC50 = 48.7 nM T87024 COZT93 44555290 IC50 = 45.3 nM T87024 CF52AX 44561723 Ki = 4 nM T87024 C30KHR 44571366 EC50 = 23200 nM T87024 C65RAJ 45102601 IC50 > 10000 nM T87024 COE8U0 45267045 IC50 = 1540 nM T87024 CIU59L 45485172 Ki = 2.9 nM T87024 CK54YN 45485173 Ki = 4.4 nM T87024 CC0FZ7 45485177 Ki = 2.22 nM T87024 CTH4K5 45485188 Ki = 6 nM T87024 CAGV92 45485189 Ki = 7.5 nM T87024 CBDN87 45485190 Ki = 18.5 nM T87024 CH40SO 45485194 Ki = 12.2 nM T87024 CO4EW7 45485195 Ki = 63 nM T87024 CL53EJ 45485210 Ki = 8.2 nM T87024 CWAF36 45485215 Ki = 9 nM T87024 C3OY6C 46207982 Ki = 0.2 nM T87024 CGNR92 46207983 Ki = 0.3 nM T87024 CY9O4P 46225190 EC50 = 1030 nM T87024 CW1DK8 46227020 Ki = 3.91 nM T87024 C0V8GA 46230999 Ki = 7.6 nM T87024 CSQ05T 46231000 Ki = 4.1 nM T87024 CQ0PG3 46231001 Ki = 3.8 nM T87024 C7JUX8 46231002 Ki = 0.9 nM T87024 CUM25P 46231003 Ki = 16.3 nM T87024 CS39BZ 46231004 Ki = 19.7 nM T87024 C1B7JZ 46835756 IC50 = 100000 nM T87024 CXM1F2 46849915 IC50 = 1100 nM T87024 C4J2RY 46849917 IC50 = 1600 nM T87024 C1JYR0 46849919 IC50 = 3300 nM T87024 CCR1A3 46850086 IC50 = 3400 nM T87024 C2VFJ3 46850257 IC50 = 800 nM T87024 CGV26A 46881557 IC50 = 35 nM T87024 CTWN14 46881596 IC50 = 45 nM T87024 CY5C3U 46881597 IC50 = 66 nM T87024 C27EWN 46881598 IC50 = 60 nM T87024 CI7V8T 46881599 IC50 = 33 nM T87024 C4UOK5 46884581 EC50 = 11800 nM T87024 CH42JI 46884664 EC50 = 190 nM T87024 CP9QX3 46905980 Ki = 6.8 nM T87024 C0G8IQ 49851437 Ki = 20.4 nM T87024 CL5KM1 50942504 Ki = 6 nM T87024 C9YJ6I 51002649 Ki = 3.5 nM T87024 CU8DB9 52108098 IC50 = 2200 nM T87024 CI8MR7 52108102 IC50 = 930 nM T87024 CBN28M 52108104 IC50 = 13100 nM T87024 C8CN5R 52108106 IC50 = 6800 nM T87024 CJNB60 52108120 IC50 = 14900 nM T87024 C7QPU6 52110752 IC50 = 5700 nM T87024 CD52WQ 52111959 IC50 = 790 nM T87024 C01HRY 52911915 IC50 = 25000 nM T87024 CS3CP8 52911916 IC50 = 35000 nM T87024 CJ25OX 52911966 IC50 = 13000 nM T87024 C0WK3Q 53016260 IC50 > 25000 nM T87024 CQ7H2G 53239243 IC50 = 2200 nM T87024 CNFJ51 53239460 IC50 = 3000 nM T87024 CHM51G 53251303 IC50 = 1900 nM T87024 C98JVW 53318054 Ki = 13.7 nM T87024 C8ALJ5 53319397 Ki = 325.8 nM T87024 C1FNQ2 53378106 IC50 = 5300 nM T87024 C1QRG2 53493644 IC50 = 24000 nM T87024 CV8JY1 53493648 IC50 = 25600 nM T87024 CZQ82K 53493779 IC50 = 24000 nM T87024 CZ1BM9 53493913 IC50 = 42000 nM T87024 CW9I0A 53493914 IC50 = 30000 nM T87024 CNCT04 53493915 IC50 = 25000 nM T87024 C0RGT1 53494038 IC50 = 48000 nM T87024 C7W1DF 53494458 IC50 = 17800 nM T87024 CQ0G6F 53494589 IC50 = 26600 nM T87024 CIV64S 53494953 Ki = 2.1 nM T87024 C3WS1P 54579968 IC50 = 58 nM T87024 C30GEJ 54579969 IC50 = 19 nM T87024 C2YET3 54579970 IC50 = 85 nM T87024 C5D2QO 54581518 Ki = 2.8 nM T87024 CNUM69 54584466 IC50 = 58 nM T87024 CJ2M1Z 54584903 IC50 = 182 nM T87024 C0JE4A 54585860 IC50 = 204 nM T87024 CV59YQ 54587360 IC50 = 75 nM T87024 C1HC0W 54612009 IC50 = 3300 nM T87024 C27ZMD 56849564 Ki = 3.86 nM T87024 C5B1EG 56850124 Ki > 1000 nM T87024 CH41IQ 56851172 Ki = 71.2 nM T87024 CK6U2R 56851599 Ki = 3.24 nM T87024 C5V7ZA 56851600 Ki = 7.71 nM T87024 C90MUF 57176479 Ki = 4672 nM T87024 CZ1T2S 57342784 IC50 = 4800 nM T87024 C6QC5O 57342787 IC50 = 14900 nM T87024 CIKX89 57342788 IC50 = 7800 nM T87024 C9FQD4 57396865 Ki = 11.4 nM T87024 C5A2HZ 57494778 Ki = 79.4 nM T87024 CTA24H 57578199 IC50 < 410 nM T87024 C9RA3F 57604425 IC50 > 50000 nM T87024 CVYT50 58220153 IC50 = 102 nM T87024 CS4AT1 58230640 IC50 = 280000 nM T87024 CEM3I4 58230686 IC50 = 240000 nM T87024 CS12RF 58446617 EC50 = 14900 nM T87024 CI2R4E 58468753 IC50 = 250 nM T87024 CH52UI 58469732 IC50 = 170 nM T87024 C2AV1Y 58469766 IC50 = 270 nM T87024 C1D9IN 58512317 IC50 = 23800 nM T87024 C7OTM1 58512491 IC50 = 15300 nM T87024 CC8ZH7 58660303 IC50 = 7100 nM T87024 CU1D5F 58795397 Ki = 260.4 nM T87024 C1OBH0 59264348 IC50 = 3700 nM T87024 CWZ1C3 60085496 EC50 = 21900 nM T87024 C2B0NS 60172115 IC50 = 100 nM T87024 CJV35M 63531802 Ki = 48.98 nM T87024 CNJT32 65476810 Ki = 112.2 nM T87024 CQ4W1V 65476811 Ki = 2818.38 nM T87024 COYR57 65476812 Ki = 385.6 nM T87024 CP2U6L 65477722 Ki = 47.86 nM T87024 CZ95NY 65479031 Ki = 12 nM T87024 CZJ29C 65479234 Ki = 21.88 nM T87024 CRXJ18 65489139 Ki = 117.49 nM T87024 CP6DJ9 65489343 Ki = 891.25 nM T87024 C4DJ3X 65489349 Ki = 524.81 nM T87024 C5R8ZY 65489731 Ki = 18.62 nM T87024 C2YST5 65490532 Ki = 5128.61 nM T87024 CA7M4I 65490730 Ki = 24.3 nM T87024 C3VU9X 65491716 Ki = 130.6 nM T87024 C06MOJ 65498771 Ki = 1023.29 nM T87024 CC8S4B 65498772 Ki = 1534.7 nM T87024 C14MAI 65501638 Ki = 407.38 nM T87024 CQU9W0 66556402 Ki = 40 nM T87024 CJ4R7E 66571561 IC50 = 1200 nM T87024 CI3M7H 67336827 IC50 = 1100 nM T87024 CIFP45 68360006 IC50 = 17000 nM T87024 CC7TH2 68540305 IC50 > 100000 nM T87024 C9JMF7 68551830 IC50 = 1600 nM T87024 CXS67Z 68552247 IC50 = 920 nM T87024 CWE58F 68553100 IC50 = 5400 nM T87024 CH54DU 68553676 IC50 = 1300 nM T87024 CY8HE3 68553756 IC50 = 590 nM T87024 C1LYJ4 68553873 IC50 > 10000 nM T87024 CAG5N8 68554590 IC50 = 760 nM T87024 CSQ53N 68555084 IC50 = 2100 nM T87024 CEI5O1 68555350 IC50 = 1100 nM T87024 CNCS47 68556083 IC50 = 930 nM T87024 CN2QL6 68556085 IC50 = 1800 nM T87024 C0TBS4 68626091 IC50 = 2100 nM T87024 CG79ML 69007129 IC50 > 50000 nM T87024 C3QH1C 70283950 IC50 = 13600 nM T87024 C4IT6K 70681870 Ki = 2.3 nM T87024 C2G3FC 70682007 IC50 = 124 nM T87024 C8T0CF 70684124 IC50 = 14 nM T87024 CKSA05 70686264 IC50 = 395 nM T87024 C14AGY 70686265 IC50 = 33 nM T87024 C0BI9A 70686266 IC50 = 32 nM T87024 CR4VM9 70686684 Ki = 5057 nM T87024 C2ZQ5R 70688384 IC50 = 19 nM T87024 CD1PU4 70688786 Ki = 31 nM T87024 CSJ2W3 70690268 Ki = 468 nM T87024 CM0N7W 70690403 IC50 = 44 nM T87024 C8FL3M 70690404 IC50 = 32 nM T87024 CG7Z2B 70694624 IC50 = 98 nM T87024 C74VAU 70696664 IC50 = 66 nM T87024 CZ3QF7 70697093 Ki = 116 nM T87024 C7MPQ3 71288593 IC50 = 110 nM T87024 CW1UG2 71288611 IC50 = 130 nM T87024 CL3E4J 71288616 IC50 = 140 nM T87024 CP89XV 71288634 IC50 = 170 nM T87024 CM8L7K 71288636 IC50 = 210 nM T87024 C5ARM6 71288638 IC50 = 86 nM T87024 C9MT0N 71288690 IC50 = 91 nM T87024 COL56G 71288696 IC50 = 100 nM T87024 C29CFW 71288697 IC50 = 68 nM T87024 CD7R9M 71288713 IC50 = 86 nM T87024 CPQ95B 71288715 IC50 = 110 nM T87024 CNC5Z3 71288739 IC50 = 120 nM T87024 C0QOF3 71288752 IC50 = 120 nM T87024 CW31HT 71288754 IC50 = 120 nM T87024 C5L4QY 71289532 IC50 = 210 nM T87024 CD0W3S 71289591 IC50 = 110 nM T87024 CSR76F 71450651 IC50 = 250 nM T87024 COV3I2 71455716 IC50 > 1000 nM T87024 CU5NQ6 71459371 IC50 > 1000 nM T87024 CZUX40 71459373 IC50 = 32.5 nM T87024 CEZ68R 71459716 IC50 = 400 nM T87024 CW1X7I 71461437 IC50 = 270 nM T87024 CX3D6F 71567514 IC50 = 2700 nM T87024 C8V6RG 71575088 Ki = 353 nM T87024 CZTH21 71575184 Ki = 121 nM T87024 CJKE41 71575185 Ki = 13.8 nM T87024 CZP06J 71575186 Ki = 83.5 nM T87024 C1R8UM 71575298 Ki = 28.9 nM T87024 CR1O2S 71575299 Ki = 39.2 nM T87024 C7N4RG 71575300 Ki > 10000 nM T87024 CN1X5W 71602710 IC50 = 36000 nM T87024 CK5PY7 71602711 IC50 = 29000 nM T87024 CJ2H4C 71602712 IC50 = 6500 nM T87024 C3RF1G 71602714 IC50 = 4000 nM T87024 CBGZ04 71602715 IC50 = 5000 nM T87024 C5VN6X 71602759 IC50 = 36000 nM T87024 CXJ01L 71712418 Ki = 1097.8 nM T87024 C07TGH 71714506 Ki = 31.5 nM T87024 CL7P0R 71764197 Ki = 111 nM T87024 CSU48O 71764198 Ki = 1180 nM T87024 CZ40WM 71764199 Ki = 758 nM T87024 C0FP6I 71764227 IC50 = 12200 nM T87024 C9K4SL 71764228 IC50 = 10660 nM T87024 CY37SI 71764366 Ki = 0.895 nM T87024 CK4W0J 71764367 Ki = 242 nM T87024 CAQC08 71764368 Ki = 15.7 nM T87024 CG4PR6 71764406 IC50 = 7560 nM T87024 CBT6S2 71764617 IC50 = 13070 nM T87024 CSG6M3 71764618 IC50 = 10320 nM T87024 C48RMB 71764619 IC50 = 18350 nM T87024 C2A5CJ 71764828 IC50 = 10220 nM T87024 CJ7OI3 71764829 IC50 = 7870 nM T87024 C5G7AJ 71764830 IC50 = 7060 nM T87024 CI4Q6K 71764831 IC50 = 6510 nM T87024 CBX6Q9 71764832 IC50 = 14160 nM T87024 CTSK68 71811225 IC50 = 9500 nM T87024 C1K6OW 71811226 IC50 = 18100 nM T87024 CU3N9R 71811227 IC50 = 18400 nM T87024 CS2L4B 71811228 IC50 = 7400 nM T87024 CL4DT9 71811229 IC50 = 5500 nM T87024 CHR8V0 71811259 IC50 = 6800 nM T87024 C0MV3O 71811291 IC50 > 50000 nM T87024 C7UYD4 71811292 IC50 > 50000 nM T87024 C7XL3N 71811293 IC50 > 50000 nM T87024 CQC8D1 71816462 Ki = 0.895 nM T87024 CFIX39 72192258 IC50 = 3960 nM T87024 CP9X1F 72205031 IC50 = 23800 nM T87024 CJ0Q1P 72205032 IC50 = 14600 nM T87024 C2FKW5 72205033 IC50 = 2200 nM T87024 CMDA21 72205034 IC50 = 5900 nM T87024 C2F6QU 72205035 IC50 = 3200 nM T87024 CHB14T 72205211 IC50 = 19900 nM T87024 CJ3N9O 72205212 IC50 = 15900 nM T87024 CVJY89 72205213 IC50 = 19100 nM T87024 C0ZR3O 72205214 IC50 = 18900 nM T87024 CZ9ED0 72205215 IC50 = 20100 nM T87024 C1LIK8 72205216 IC50 = 8300 nM T87024 C7I4MU 72205404 IC50 = 17800 nM T87024 CDY89J 72205405 IC50 = 7300 nM T87024 CR7TP1 72205406 IC50 = 10100 nM T87024 C1K4TV 72205407 IC50 = 13300 nM T87024 C78YAO 72205408 IC50 = 5800 nM T87024 CCES98 72205409 IC50 = 10900 nM T87024 CIXJ32 72205410 IC50 = 10500 nM T87024 CRGI65 72205594 IC50 = 19100 nM T87024 CJ2FW4 72205595 IC50 = 12500 nM T87024 C45BXP 72543919 IC50 = 4830 nM T87024 C78ZPH 72544154 IC50 = 8180 nM T87024 CKAG40 72544155 IC50 = 3110 nM T87024 CPH96F 72544156 IC50 = 6110 nM T87024 CTW28Y 72544382 IC50 = 6880 nM T87024 C6TQ7M 72545286 IC50 = 4770 nM T87024 CBL6J5 72545287 IC50 = 4430 nM T87024 C9ZB1M 72725489 IC50 = 51000 nM T87024 CLVB69 73294880 IC50 > 10000 nM T87024 CGZK85 73296378 IC50 = 7 nM T87024 C9L3VR 73296809 IC50 = 32 nM T87024 C2S9PZ 73296810 IC50 = 18 nM T87024 C4XR1C 73297137 IC50 = 6 nM T87024 CCPI94 73297139 IC50 = 123 nM T87024 C4W7LS 73345877 IC50 = 100000 nM T87024 CTUQ90 73346005 Ki > 242 nM T87024 CCS12L 73346452 IC50 = 17300 nM T87024 C38OPD 73347953 IC50 = 9800 nM T87024 CU9FP1 73347954 IC50 = 13200 nM T87024 CLP90V 73347955 IC50 = 9600 nM T87024 C8W6DQ 73349062 Ki > 242 nM T87024 CW03TX 73350560 Ki = 116.8 nM T87024 CGSK10 73350561 Ki = 79.7 nM T87024 C4IL9R 73350636 Ki > 242 nM T87024 CLC9U3 73350637 Ki = 111 nM T87024 C4GT1B 73351048 IC50 = 13700 nM T87024 C0G7QU 73351049 IC50 = 14200 nM T87024 CE71NV 73351050 IC50 = 13500 nM T87024 C6V0CI 73351053 IC50 = 14100 nM T87024 C0P2JF 73352070 Ki = 28.4 nM T87024 CE7Q5V 73352141 IC50 = 18500 nM T87024 C7VL9F 73352527 IC50 = 14900 nM T87024 C1A6BY 73353594 Ki = 15.7 nM T87024 CY37DV 73355034 Ki = 1030.1 nM T87024 C0VW4X 73355546 IC50 = 12600 nM T87024 C0XP4S 73355547 IC50 = 16400 nM T87024 CW9X2J 73355548 IC50 = 12800 nM T87024 CXF2N4 73357092 IC50 = 4800 nM T87024 CNS32L 73357093 IC50 = 11500 nM T87024 CTJU47 73357094 IC50 = 16800 nM T87024 C37PAK 73357095 IC50 = 6500 nM T87024 CIS76V 76283251 Ki = 588.84 nM T87024 CU9P7V 76283252 Ki = 20662 nM T87024 C7FOW8 76283253 Ki = 17.6 nM T87024 C72VSC 76283256 Ki = 152.6 nM T87024 CM37BJ 76283490 Ki = 21 nM T87024 CHT45P 76283491 Ki = 118.5 nM T87024 CYJ87Q 76313138 Ki = 102.74 nM T87024 C91IXN 76318192 Ki = 9.1 nM T87024 C1Q6ZD 76325788 Ki = 13.6 nM T87024 CQ50IP 76329071 Ki = 63.57 nM T87024 C0ZFI3 76333017 Ki = 24.8 nM T87024 CR14VW 76336360 Ki = 25.54 nM T87024 CFQH52 80755129 IC50 = 80 nM T87024 CH4FK6 80765618 IC50 = 10200 nM T87024 CKYI49 80765970 IC50 = 620 nM T87024 C0CL4Y 80772460 IC50 = 2000 nM T87024 CDK40F 80773548 IC50 = 2800 nM T87024 CVB4X2 80774737 IC50 = 20600 nM T87024 CL03NW 80777722 IC50 = 3900 nM T87024 C39DIK 80777938 IC50 = 3100 nM T87024 CYBD08 80791041 IC50 = 3600 nM T87024 C8WK3D 80793928 IC50 = 580 nM T87024 CYT97P 80832588 IC50 = 1900 nM T87024 C51CLO 86279144 Ki = 84.48 nM T87024 CE9X5J 86713212 IC50 = 2500 nM T87024 C45CME 89681657 IC50 < 1000 nM T87024 C3R4PD 89970609 IC50 = 470 nM T87024 C06FNJ 89970660 IC50 = 5400 nM T87024 CE1IW4 89970765 IC50 = 610 nM T87024 CEF8J5 90040128 IC50 = 93 nM T87024 CD48HU 90277509 IC50 > 10000 nM T87024 CX28SL 90644922 IC50 = 18 nM T87024 CHD0Z7 90644923 IC50 > 10000 nM T87024 CYPJ75 90644924 IC50 = 32 nM T87024 CQ2J6Y 90654541 Ki = 244 nM T87024 C85HOG 90654542 Ki = 39.3 nM T87024 CAE28Q 90654543 Ki = 56.4 nM T87024 CWF6X2 90654981 IC50 = 24200 nM T87024 C1PY0T 90676323 IC50 = 4400 nM T87024 CZ5BG2 101423563 IC50 > 50000 nM T87024 C6W2JF 101898808 IC50 > 100000 nM T87024 C4BD5S 102115496 IC50 = 15900 nM T87024 CTL20G 102196384 IC50 > 10000 nM T87024 C0O9XI 102259962 IC50 > 100000 nM T87024 C5PBW3 102398558 IC50 > 10000 nM T87024 CAS5M1 102407747 IC50 > 50000 nM T87024 CO71AT 117809085 EC50 = 11400 nM T87024 C1J0IZ 118711805 IC50 > 100000 nM T87024 CJG10W 118711813 IC50 = 5000 nM T87024 C2Q8IE 118711815 IC50 = 24200 nM T87024 C9U5SV 118712170 IC50 = 13400 nM T87024 C9KUS7 118712171 IC50 = 6100 nM T87024 C5W7PM 118713185 IC50 = 1500 nM T87024 CQ07AH 118713186 IC50 > 10000 nM T87024 C5OFH2 118713187 IC50 > 10000 nM T87024 C9ZGB4 118713188 IC50 > 10000 nM T87024 C7Z2GA 118713189 IC50 > 10000 nM T87024 C03URO 118713190 IC50 > 10000 nM T87024 CYK30H 118713191 IC50 > 10000 nM T87024 CK53ME 118713192 IC50 > 10000 nM T87024 C35IDH 118713193 IC50 < 380 nM T87024 CM7UC8 118713194 IC50 > 10000 nM T87024 C5C8LX 118713195 IC50 = 550 nM T87024 C1RH3Y 118713196 IC50 > 10000 nM T87024 C1A6TD 122164218 IC50 = 2600 nM T87024 CUML76 122179364 IC50 = 95900 nM T87024 C2ELQ6 122179365 IC50 = 28000 nM T87024 CU4J3V 122179366 IC50 = 34300 nM T87024 CG8C1U 122179367 IC50 = 71900 nM T87024 CV0J6F 122179368 IC50 = 10100 nM T87024 CLM90O 122179370 IC50 = 1200 nM T87024 CB0TP1 122179371 IC50 = 43500 nM T87024 CMX95N 122181785 IC50 = 26000 nM T87024 CMF53A 122181787 IC50 = 17000 nM T87024 CEJ29G 122181789 IC50 = 7700 nM T87024 CC82TX 122181791 IC50 = 1600 nM T87024 CLRW41 122181793 IC50 = 26000 nM T87024 CD0NU8 122181797 IC50 = 800 nM T87024 CB03DR 122182244 Ki = 94.8 nM T87024 CI6WT0 122182245 Ki = 251.5 nM T87024 C3X5KJ 122182246 Ki = 87.1 nM T87024 CT5G1Q 122182247 Ki = 139.9 nM T87024 CCT7H6 122182248 Ki = 190.2 nM T87024 CML3T5 122182249 Ki = 113.3 nM T87024 CMO1C3 122182250 Ki = 125.8 nM T87024 CIT52U 122182251 Ki = 27.6 nM T87024 C19GJH 122182252 Ki = 15.3 nM T87024 CUOB01 122182253 Ki = 37.1 nM T87024 CW2V5B 122182254 Ki = 703.3 nM T87024 C75OCP 122182255 Ki = 741 nM T87024 CVH2T0 122182256 Ki = 56 nM T87024 CKQF12 122182257 Ki = 357.9 nM T87024 C7AUF8 122182258 Ki = 129.6 nM T87024 C7BXY4 122182259 Ki = 92.4 nM T87024 CCEL74 122182260 Ki = 45.9 nM T87024 C32GEV 122182261 Ki = 84 nM T87024 CWIT38 122182262 Ki = 85.1 nM T87024 CMVS36 122182263 Ki = 107 nM T87024 CLW95X 122182264 Ki = 98.9 nM T87024 C4TNB1 122182265 Ki = 286.8 nM T87024 CQ4R0K 122182266 Ki = 50.8 nM T87024 C5C8FY 122182267 Ki = 459.5 nM T87024 C7NV9G 122182268 Ki = 36.2 nM T87024 CU3NJ6 122182269 Ki = 60 nM T87024 CS84HC 122182270 Ki = 214.2 nM T87024 C8EYO3 122182271 Ki = 235.4 nM T87024 CFV32E 122182272 Ki = 130.8 nM T87024 C1LHQ2 122182273 Ki = 138.5 nM T87024 C24PHB 122182274 Ki = 109.7 nM T87024 C1U3FZ 122182275 Ki = 264.8 nM T87024 CX5NB4 122182276 Ki = 73.6 nM T87024 CAU9H6 122182277 Ki = 129.5 nM T87024 C2RB1F 122182278 Ki = 142.4 nM T87024 CTMV35 122182279 Ki = 125.3 nM T87024 C8XU3B 122191852 IC50 = 15000 nM T87024 CW1ID8 126512451 Ki = 770.1 nM T87024 CSA9G5 127025485 Ki = 437.9 nM T87024 C7CF1O 127026387 Ki = 191.1 nM T87024 C43JRQ 127027320 Ki = 25.7 nM T87024 CJN7U9 127028024 Ki = 357.7 nM T87024 CM87CX 127030059 Ki = 6.82 nM T87024 CKW7U0 127037724 EC50 > 300000 nM T87024 CCW3V2 127037725 EC50 > 300000 nM T87024 CK57HV 127037726 EC50 > 300000 nM T87024 CR14WP 127037731 EC50 = 97900 nM T87024 C7J1FZ 127037732 EC50 = 105200 nM T87024 CSAB54 127037733 IC50 = 203700 nM T87024 CKEW84 127037734 EC50 = 65400 nM T87024 CXUM93 127037767 IC50 = 2900 nM T87024 CSXQ94 127037768 IC50 = 3400 nM T87024 CVH0L5 127037769 IC50 = 3900 nM T87024 CFBI32 127037770 IC50 = 19600 nM T87024 CU5D2R 127038083 EC50 > 300000 nM T87024 CP2GI5 127038098 IC50 > 50000 nM T87024 CA8V7Z 127038099 IC50 = 4000 nM T87024 CBY32I 127038456 EC50 = 89900 nM T87024 CMT6N9 127039696 IC50 > 50000 nM T87024 C0XJS3 127039805 IC50 = 4000 nM T87024 CIBU28 127041690 IC50 = 16800 nM T87024 C2TZ4U 127041980 IC50 > 50000 nM T87024 CEF8N6 127042668 IC50 = 5600 nM T87024 CY05OR 127045901 IC50 = 71.28 nM T87024 CYJ56A 127045902 IC50 = 22.54 nM T87024 CX6SU5 127045903 IC50 = 51.81 nM T87024 C50ZPS 127045904 IC50 = 45.29 nM T87024 C39PUO 127046118 IC50 = 77.45 nM T87024 C9LF7P 127047722 IC50 = 45.88 nM T87024 CZ3PT1 127047832 IC50 = 46.12 nM T87024 CQ2TI9 127047833 IC50 = 51.77 nM T87024 C0EO6S 127047834 IC50 = 38.96 nM T87024 C0GQ9Z 127047951 IC50 = 55.86 nM T87024 CC7M1B 127047952 IC50 = 30.74 nM T87024 CQ3O4A 127047953 IC50 = 65.5 nM T87024 C9SCI6 127047954 IC50 = 37.36 nM T87024 C0O4AZ 127047955 IC50 = 17.36 nM T87024 CGM1Y0 127047956 IC50 = 49.14 nM T87024 CC64LO 127048346 IC50 > 25000 nM T87024 CY48DV 127048347 IC50 = 2300 nM T87024 C7F6LR 127048348 IC50 = 1500 nM T87024 CX3K0P 127048349 IC50 = 1700 nM T87024 C85UWQ 127048350 IC50 = 11300 nM T87024 C5C1JP 127048771 IC50 = 10110 nM T87024 C3XBG6 127049292 IC50 = 12500 nM T87024 C5KJQ6 127049344 IC50 > 25000 nM T87024 C2W5QI 127049933 IC50 = 5900 nM T87024 CVR3N2 127050660 IC50 = 9200 nM T87024 C4JMF5 127050661 IC50 = 11750 nM T87024 CV0HR8 127050925 IC50 = 3500 nM T87024 CCOK39 127050926 IC50 = 1900 nM T87024 CLH53U 127051777 IC50 > 25000 nM T87024 C6U0PH 127051778 IC50 > 25000 nM T87024 C3PEZ8 127052081 IC50 > 25000 nM T87024 CLH6T3 132547257 IC50 = 66360 nM T87024 CS21FU 132934435 IC50 = 2700 nM T87024 CPJ8I0 132934436 IC50 = 8400 nM T87024 CO54NG 134133007 IC50 = 520 nM T87024 C2JA7H 134140987 IC50 = 7400 nM T87024 C2E1WL 134142133 IC50 = 10900 nM T87024 CFM92E 134143791 IC50 = 9900 nM T87024 C6Q9WM 134145849 IC50 = 12200 nM T87024 CJ6W1Y 135582041 IC50 = 500 nM T87024 CHMW08 135582042 IC50 = 2300 nM T87024 CFW83Z 135693450 IC50 = 800 nM T87024 CTMC18 135693451 IC50 = 1100 nM T87024 C8Y1CP 135693469 IC50 = 1100 nM T87024 CCF4D1 135693470 IC50 = 1700 nM T87024 C6RA8X 135693471 IC50 = 1400 nM T87024 CYUB25 135693472 IC50 = 1900 nM T87024 C1XQY2 135923992 IC50 = 138 nM T87024 C76ORP 135937123 IC50 = 3200 nM T87024 CNA50S 135937129 IC50 = 3700 nM T87024 CN3EF7 135995955 IC50 = 4300 nM T87024 C0UR9T 135995956 IC50 = 15800 nM T87024 C3VA4S 135995957 IC50 = 1300 nM T87024 CQ5BX7 135995958 IC50 = 2900 nM T87024 CBL8M1 136264407 Ki = 34.72 nM T87024 C78ZBO 136276907 IC50 = 44 nM T87024 CK6C8S 136286700 IC50 = 8500 nM T87024 C6GM9U 137632892 IC50 = 15380 nM T87024 CO1FZ2 137636537 IC50 = 18970 nM T87024 CV8W7S 137637059 IC50 = 1900 nM T87024 C2WBP4 137637064 IC50 = 1400 nM T87024 CZ5WE1 137637732 IC50 = 8300 nM T87024 CC7E4I 137638765 IC50 = 1000 nM T87024 CR5G9J 137638769 IC50 = 3800 nM T87024 CQXF56 137639807 IC50 = 2300 nM T87024 C23OHG 137640005 IC50 = 16500 nM T87024 CUA7O1 137641177 IC50 = 23390 nM T87024 CS4X7J 137641292 IC50 = 10720 nM T87024 CQ8B9C 137641449 IC50 = 7200 nM T87024 C3EL4I 137642431 IC50 = 4900 nM T87024 CVW3C9 137643867 IC50 = 12480 nM T87024 CC2SY8 137646193 IC50 = 13300 nM T87024 CZU89F 137646680 IC50 = 7800 nM T87024 C9J3XC 137647729 IC50 = 4400 nM T87024 CJP1G6 137648183 IC50 = 1700 nM T87024 C7Z4MI 137649813 IC50 = 2900 nM T87024 CXO54P 137650485 IC50 = 19440 nM T87024 CSN3M6 137652664 IC50 = 21760 nM T87024 CSO97E 137653574 IC50 = 6600 nM T87024 CB2DR3 137654189 IC50 = 29220 nM T87024 CZME36 137654357 IC50 = 11200 nM T87024 C0LR3F 137654627 IC50 = 3100 nM T87024 CT51VW 137658213 IC50 = 4300 nM T87024 COL58K 137659202 IC50 = 8300 nM T87024 CU6D3I 137660068 IC50 = 10400 nM T87024 CA6O8X 137660402 IC50 = 8940 nM T87024 C31MDX 137661164 IC50 = 14400 nM T87024 C2XLH1 145949548 IC50 = 23800 nM T87024 C3X0BF 145951162 IC50 = 11550 nM T87024 CRL14N 145951634 IC50 = 16290 nM T87024 CAE3F6 145952153 IC50 = 17850 nM T87024 C4SAC7 145952735 EC50 = 80100 nM T87024 CS92HK 145952951 IC50 = 23540 nM T87024 CAOK81 145954140 IC50 = 13400 nM T87024 CV8N3W 145954662 IC50 = 25000 nM T87024 CG0L8C 145955195 EC50 = 274000 nM T87024 C98ASV 145956279 IC50 = 18550 nM T87024 C9H8DN 145957368 EC50 = 54800 nM T87024 CL4V8A 145957466 IC50 = 15890 nM T87024 CQ2F9N 145958030 IC50 = 18050 nM T87024 CJM1L6 145958479 IC50 = 20720 nM T87024 C5LD0P 145958580 EC50 = 39500 nM T87024 CM9N5K 145958693 IC50 = 8280 nM T87024 CJX6Y0 145958697 IC50 = 18310 nM T87024 C6VS1G 145960818 IC50 > 100000 nM T87024 CX84UO 145960840 IC50 = 22700 nM T87024 C6BN0G 145960867 IC50 = 8700 nM T87024 C3HO6N 145967633 IC50 = 8200 nM T87024 CN2H4A 145967886 IC50 = 5640 nM T87024 CQ0U4M 145967937 IC50 = 11440 nM T87024 CIV32Q 145968088 IC50 = 4600 nM T87024 C47HPQ 145968126 IC50 = 18280 nM T87024 CTH57O 145968156 IC50 = 2500 nM T87024 C0PX2K 145968691 IC50 = 43600 nM T87024 CSR1I9 145969054 IC50 = 4100 nM T87024 CB8EM7 145969243 IC50 = 18940 nM T87024 C1L0SY 145969265 IC50 > 10000 nM T87024 C0EO1R 145969271 IC50 > 10000 nM T87024 C1ZFK2 145969492 IC50 = 16810 nM T87024 CIH43M 145969511 IC50 > 10000 nM T87024 CC4F6E 145969712 IC50 > 10000 nM T87024 C36NST 145969906 IC50 = 6600 nM T87024 CPK3D5 145970010 IC50 = 17330 nM T87024 CP3I6Z 145970131 IC50 > 10000 nM T87024 CHN96I 145970153 IC50 = 19740 nM T87024 C3AJF1 145970176 IC50 > 10000 nM T87024 C5IFR6 145970205 IC50 > 10000 nM T87024 C51AZL 145970361 IC50 = 20610 nM T87024 C20CDL 145970677 IC50 = 5050 nM T87024 CGNM74 145970882 IC50 > 10000 nM T87024 CKY16Q 145970910 IC50 = 7350 nM T87024 CM0GA5 145970919 IC50 > 10000 nM T87024 C2VKL5 145970929 IC50 > 10000 nM T87024 CJZ24V 145971052 IC50 = 22550 nM T87024 CJEQ52 145971111 IC50 > 10000 nM T87024 CQ9K7V 145972919 IC50 = 5840 nM T87024 C2G5CI 145973156 EC50 = 5930 nM T87024 C3VD1Z 145973583 IC50 = 12500 nM T87024 C1YX4W 145975729 IC50 = 10430 nM T87024 C4R3UA 145978145 IC50 = 85500 nM T87024 CFH6X2 145980202 IC50 = 17680 nM T87024 C09CGW 145987951 IC50 = 6200 nM T87024 CQ1KL7 145988407 IC50 = 8860 nM T87024 CF8TY4 145990938 IC50 = 7200 nM T87024 CZL1W8 145992158 IC50 = 8290 nM T87024 CMY0S7 145992432 IC50 = 7930 nM T87024 C74MNX 145993766 IC50 = 5920 nM T87024 CA84QP 145994000 IC50 = 17950 nM T87024 CVT98S 155510374 IC50 = 3050 nM T87024 C0IFO1 155512131 IC50 = 17440 nM T87024 CNYU38 155512854 IC50 = 9600 nM T87024 CAI92C 155513704 IC50 = 44520 nM T87024 C9ACN1 155514094 IC50 = 3630 nM T87024 CN73HA 155514383 IC50 = 3550 nM T87024 C60AEI 155517024 IC50 = 3870 nM T87024 C3HS6G 155517170 IC50 = 17890 nM T87024 C6P0YN 155517656 IC50 = 3400 nM T87024 C43LSX 155521501 IC50 = 3310 nM T87024 CZL82K 155522864 IC50 = 15720 nM T87024 C7MGP1 155524606 IC50 = 4900 nM T87024 CSX93I 155529365 IC50 = 17230 nM T87024 C2NX1W 155529394 IC50 = 3160 nM T87024 C87WTD 155531118 IC50 = 2000 nM T87024 C7HIJ5 155531717 IC50 = 21700 nM T87024 C57NLC 155532779 IC50 = 5470 nM T87024 CCAV95 155533217 IC50 = 17500 nM T87024 C2AZ1D 155534166 Ki = 6.9 nM T87024 C70XUL 155536929 IC50 = 3450 nM T87024 CPGY39 155537952 IC50 = 2310 nM T87024 C7MDN9 155538092 IC50 = 60 nM T87024 CC1W3Y 155538615 IC50 = 4600 nM T87024 CP7Y8G 155538698 IC50 = 3980 nM T87024 C9ZC1Q 155540322 IC50 = 4200 nM T87024 CD81WU 155541984 IC50 = 2800 nM T87024 C50NRO 155542946 IC50 = 8065 nM T87024 CG5OT4 155544377 IC50 = 3860 nM T87024 C1XM3K 155555566 IC50 = 2370 nM T87024 CCO2Q1 155556363 IC50 = 8900 nM T87024 COH58T 155556504 IC50 = 3710 nM T87024 C90YXU 155559099 IC50 = 2410 nM T87024 CV5NU3 155560530 IC50 = 46420 nM T87024 CC48AD 155567294 IC50 = 12600 nM T87024 C9CQD6 11301908 Ki = 15 nM T87024 D00KEP 6049 IC50 = 7700 nM T87024 D00RIX 5280443 IC50 = 23000 nM T87024 D01MMU 11708629 Ki = 1.3 nM T87024 D02BBJ 11550464 Ki = 0.7 nM T87024 D02DFT 44408965 Ki = 31.2 nM T87024 D02FZQ 3552928 Ki = 108 nM T87024 D02HCQ 1794427 IC50 = 92900 nM T87024 D02YSX 197033 EC50 = 25000000 nM T87024 D03AMR 9849669 IC50 = 200 nM T87024 D03RJH 44408693 Ki = 625 nM T87024 D03THP 44408839 Ki = 5.6 nM T87024 D03TOK 11587026 Ki = 9 nM T87024 D05CCT 4139 IC50 = 500 nM T87024 D05GRI 5354238 Ki = 54.24 nM T87024 D05PTT 5281792 EC50 = 20300 nM T87024 D06DRD 160843 Ki = 0.14 nM T87024 D06YGF 5281787 EC50 = 8410 nM T87024 D07LFZ 21788024 Ki = 6.1 nM T87024 D07SNW 11537013 Ki = 837 nM T87024 D08GKL 11632242 Ki = 22.6 nM T87024 D08TME 4373578 Ki = 185 nM T87024 D09MQZ 44408738 Ki = 6.1 nM T87024 D09RAM 44408840 Ki = 9.6 nM T87024 D09SOY 15054176 EC50 = 4170 nM T87024 D09UWI 14905189 Ki = 4 nM T87024 D0A1CM 5281855 IC50 = 100000 nM T87024 D0B1CL 11579589 Ki = 2.3 nM T87024 D0C1AU 6177872 Ki = 500 nM T87024 D0C9QW 11543378 Ki = 2.8 nM T87024 D0F5EJ 11375002 IC50 = 45000 nM T87024 D0G3TK 5280863 IC50 = 75100 nM T87024 D0H0AT 10425576 Ki = 18.5 nM T87024 D0I8XD 10013901 Ki = 1.2 nM T87024 D0I9NH 11499570 Ki = 11.5 nM T87024 D0L7MD 466289 Ki = 29 nM T87024 D0M4IE 9549196 IC50 = 8400 nM T87024 D0NJ4H 5281670 IC50 = 30300 nM T87024 D0O5FK 10171487 Ki = 0.87 nM T87024 D0P0CB 11574659 Ki = 13.2 nM T87024 D0R0LQ 11673398 Ki = 12 nM T87024 D0R4FM 122850 IC50 > 500000 nM T87024 D0T2QL 444539 IC50 > 100000 nM T87024 D0T3PW 5281672 IC50 < 3000 nM T87024 D0U6KE 11507217 Ki = 9 nM T87024 D0V9EN 689043 EC50 = 216000 nM T87024 D0W0WL 11608986 Ki = 7.5 nM T87024 D0X1EY 11703303 Ki = 72.5 nM T87024 D0Y7HG 5281616 IC50 > 500000 nM T87024 D0Z7EL 5280647 IC50 < 3000 nM T97196 D0B3HD 2519 IC50 = 200000 nM T97196 D02NUT 15953870 IC50 = 6 nM T97196 D06DMQ 59472121 Ki = 44 nM T97196 D0H9DA 54761306 IC50 > 30000 nM T97196 D0O1IM 58298318 IC50 > 30000 nM T97196 D0VF6E 1401 IC50 = 17600 nM T97196 D0VG0D 11977753 IC50 = 7 nM T97196 D0W7HE 56649450 IC50 > 10000 nM T97196 D0XD4I 118502708 IC50 = 0.57 nM T97196 D09SFV 3973 IC50 > 10000 nM T97196 CAUK86 108130 IC50 = 1740000 nM T97196 CG53MZ 277839 IC50 = 250 nM T97196 C3V1HN 1490241 IC50 > 40000 nM T97196 CJ19SK 2723790 IC50 = 200 nM T97196 C87VQB 5353854 IC50 = 12000 nM T97196 CJ61TH 9817584 IC50 = 600 nM T97196 CKAD93 11433009 IC50 = 3 nM T97196 C1SNR6 13141222 IC50 > 8000 nM T97196 C2AXJ7 16203250 IC50 > 10000 nM T97196 CAI9S5 16203254 IC50 > 10000 nM T97196 C1I8YQ 16203357 IC50 > 10000 nM T97196 CGQ82D 16203358 IC50 > 100000 nM T97196 C9E4OH 16203360 IC50 > 100000 nM T97196 C42FYM 16203361 IC50 = 28500 nM T97196 CN7QP8 16203467 IC50 = 10000 nM T97196 CR2S5J 16203591 IC50 > 10000 nM T97196 CD4XG7 16203592 IC50 > 10000 nM T97196 C3FWM9 16203595 IC50 > 100000 nM T97196 CGO9N1 16203602 IC50 > 100000 nM T97196 CED0M3 16203716 IC50 > 100000 nM T97196 C79JLP 16203721 IC50 > 10000 nM T97196 C5J7FQ 16203836 IC50 > 10000 nM T97196 C2JA8F 16203837 IC50 > 100000 nM T97196 CQ1Z0V 16203940 IC50 > 100000 nM T97196 C45LZB 16203944 IC50 > 10000 nM T97196 C41EGR 16203945 IC50 > 10000 nM T97196 C4SJX6 16203947 IC50 = 4300 nM T97196 C7TOJ8 16203948 IC50 > 10000 nM T97196 CODI71 16204048 IC50 > 100000 nM T97196 CV6P2N 19088789 IC50 > 100000 nM T97196 CH3L9P 44551660 IC50 = 20 nM T97196 C3VRO9 44557921 IC50 > 10000 nM T97196 CU5K1G 46834296 IC50 > 8000 nM T97196 CM73PR 46834571 IC50 > 8000 nM T97196 CTO5B6 46834572 IC50 = 6600 nM T97196 CRJ5W8 51358113 EC50 = 28 nM T97196 CA50HJ 52915004 IC50 > 8000 nM T97196 C5R2AH 52937148 IC50 > 8000 nM T97196 CLH8Y5 52937149 IC50 > 8000 nM T97196 CT7X9U 52937150 IC50 > 8000 nM T97196 C12GTQ 52937251 IC50 > 8000 nM T97196 CQ85UH 52937252 IC50 > 8000 nM T97196 CP91TZ 52937253 IC50 = 320 nM T97196 C1MIR4 52937254 IC50 = 3000 nM T97196 CID2E8 52937255 IC50 > 8000 nM T97196 C2H9JY 52937257 IC50 > 8000 nM T97196 CPY82U 52937258 IC50 > 8000 nM T97196 C27QNB 52937357 IC50 > 8000 nM T97196 CFJB79 52937358 IC50 > 8000 nM T97196 CT5K9L 52937359 IC50 > 8000 nM T97196 C85FTW 52937360 IC50 > 8000 nM T97196 CGLT04 52937361 IC50 > 8000 nM T97196 C2ISM3 52937362 IC50 > 8000 nM T97196 C6Q2EN 52937363 IC50 > 8000 nM T97196 CFT9H6 52937453 IC50 > 8000 nM T97196 C4C6DF 52937454 IC50 > 8000 nM T97196 C0T8KI 52937455 IC50 = 2900 nM T97196 CK30PU 52937456 IC50 = 2600 nM T97196 CJU30Y 52937457 IC50 > 8000 nM T97196 C4RJB2 52937458 IC50 > 8000 nM T97196 C69SEB 52937459 IC50 > 8000 nM T97196 CPR6W2 52937553 IC50 > 8000 nM T97196 CQP02L 52937554 IC50 > 8000 nM T97196 CAHU94 52937555 IC50 > 8000 nM T97196 CQ2NU7 52937556 IC50 > 8000 nM T97196 CATX20 52937557 Ki = 4000 nM T97196 CB9WS5 52937558 IC50 = 5400 nM T97196 CUY01F 52937559 IC50 = 6600 nM T97196 CTM68E 52937659 IC50 > 8000 nM T97196 C7G9KF 52937660 IC50 > 8000 nM T97196 C5G6YD 52937661 IC50 = 5000 nM T97196 C6R5OE 52937662 IC50 > 8000 nM T97196 CDHT14 52937663 IC50 = 380 nM T97196 C0IJZ8 52937664 IC50 = 840 nM T97196 CGW25Q 52937665 IC50 = 720 nM T97196 CL04GS 52937759 IC50 = 120 nM T97196 C0Y9ZG 54761473 IC50 > 30000 nM T97196 C1YTI8 59472018 Ki > 10000 nM T97196 C76CVG 59472034 Ki = 190 nM T97196 C1EW0H 59472203 Ki = 93 nM T97196 C0MJ3L 59472343 Ki = 115 nM T97196 CI1HO0 71521971 Ki = 1300 nM T97196 CI2J9Q 71521995 Ki > 4000 nM T97196 CKB86I 71537083 Ki = 189 nM T97196 CAVL54 71554734 Ki > 10000 nM T97196 CLO1P5 72199292 IC50 > 36 nM T97196 CHX2Z3 90435584 Ki = 47 nM T97196 C05LQH 118498627 IC50 = 1.5 nM T97196 CXCF46 118498683 IC50 = 0.78 nM T97196 CJA07S 118498727 IC50 = 0.25 nM T97196 CG6D1J 118498935 IC50 = 0.33 nM T97196 CXR46C 118499887 IC50 = 0.25 nM T97196 CFVN15 118500050 IC50 = 0.24 nM T97196 CY9NW0 118500097 IC50 = 0.17 nM T97196 CXEI18 118500108 IC50 = 0.76 nM T97196 CL2Z5Y 118502821 IC50 = 2.6 nM T97196 CVY64N 118502892 IC50 = 1.1 nM T97196 CO20ET 118502895 IC50 = 0.2 nM T97196 CU1X3H 118502919 IC50 = 0.94 nM T97196 CRAF61 118523357 IC50 = 0.29 nM T97196 C5P7VH 118523411 IC50 = 1.1 nM T97196 CD0EY5 118523423 IC50 = 1.2 nM T97196 CF5HV8 118720613 IC50 = 130 nM T97196 C2UIB7 118720614 IC50 = 14000 nM T97196 CSH50J 118720615 IC50 = 4300 nM T97196 C9SF2E 118720891 IC50 = 15000 nM T97196 C4M1VF 127025043 IC50 > 40000 nM T97196 C3EJ9F 127025044 IC50 > 40000 nM T97196 C32IFD 127025045 IC50 > 40000 nM T97196 CO2F9Q 127025046 IC50 > 40000 nM T97196 C4I9VW 127025047 IC50 = 10100 nM T97196 C0GN5W 127025057 IC50 > 40000 nM T97196 C1W0BF 127025331 IC50 = 2200 nM T97196 CTV81N 127025332 IC50 > 40000 nM T97196 C3HS4B 127025333 IC50 = 6600 nM T97196 CH97GA 127025334 IC50 = 6100 nM T97196 CO27MB 127025335 IC50 = 2700 nM T97196 CR3U9D 127025341 IC50 = 1700 nM T97196 CJPU49 127025342 IC50 = 1600 nM T97196 CU4HL1 127025343 IC50 = 5300 nM T97196 CJ8HV3 127025344 IC50 = 1700 nM T97196 CJ9GV0 127025345 IC50 = 900 nM T97196 CN6Z5I 127025362 IC50 = 2100 nM T97196 CYK5C6 127025363 IC50 = 5300 nM T97196 C6HSB4 127025364 IC50 = 13300 nM T97196 CM1V6D 127025365 IC50 = 1600 nM T97196 CSAV12 127025618 IC50 = 5600 nM T97196 CVS1E5 127025637 IC50 = 800 nM T97196 CG64FH 127025644 IC50 = 1200 nM T97196 C5A1CI 127025914 IC50 = 6.3 nM T97196 CJLX39 127025921 IC50 = 800 nM T97196 CJ3ZG4 127025922 IC50 = 800 nM T97196 C4AL7I 127025923 IC50 = 1000 nM T97196 C54QBO 127025931 IC50 > 40000 nM T97196 C27DFR 127026195 IC50 = 28600 nM T97196 CL0Q2Y 127026196 IC50 = 23500 nM T97196 CJ3T8O 127026197 IC50 = 1900 nM T97196 C51JZI 127026507 IC50 = 2900 nM T97196 CXE3H1 127026831 IC50 > 40000 nM T97196 C3N6ZT 127026832 IC50 > 40000 nM T97196 CYO16P 127027754 IC50 > 40000 nM T97196 C0EQX6 127027768 IC50 > 40000 nM T97196 CO17SP 127027769 IC50 > 40000 nM T97196 CY6U1L 127027770 IC50 > 40000 nM T97196 CGRA75 127027771 IC50 = 8600 nM T97196 CC19SZ 127037860 IC50 > 40000 nM T97196 CE8Y4M 127037868 IC50 = 12500 nM T97196 CPT39E 127038233 IC50 = 2300 nM T97196 C14EHC 127038522 IC50 > 40000 nM T97196 C4OBY6 127038551 IC50 > 40000 nM T97196 CYXV95 127038563 IC50 = 2400 nM T97196 C38JYR 127039200 IC50 = 12600 nM T97196 CUY69A 127039219 IC50 = 2000 nM T97196 CZL62I 127039548 IC50 = 1200 nM T97196 CC71GK 127039891 IC50 > 40000 nM T97196 C1Z4NO 127039892 IC50 = 16900 nM T97196 CQVC56 127039893 IC50 > 40000 nM T97196 C1K6ZB 127039894 IC50 > 40000 nM T97196 C0TO7P 127039895 IC50 > 40000 nM T97196 C0KHO1 127039896 IC50 = 15000 nM T97196 CT0D2L 127039897 IC50 = 5000 nM T97196 C52JVW 127040212 IC50 > 40000 nM T97196 CX5B6Y 127040213 IC50 > 40000 nM T97196 CEZ3N0 127040541 IC50 > 40000 nM T97196 CV5UC6 127040542 IC50 > 40000 nM T97196 C6YIL9 127040543 IC50 > 40000 nM T97196 C4PK0I 127040544 IC50 = 31100 nM T97196 CZ3A2N 127040545 IC50 > 40000 nM T97196 CN12MH 127041181 IC50 > 40000 nM T97196 CYK8U7 127041513 IC50 > 40000 nM T97196 CXTS09 127041514 IC50 > 40000 nM T97196 CFT54M 127042439 IC50 = 20600 nM T97196 C17EZQ 127042473 IC50 > 40000 nM T97196 C2BU4P 127042474 IC50 > 40000 nM T97196 CNIK04 127042475 IC50 > 40000 nM T97196 C4T9SU 127042476 IC50 > 40000 nM T97196 CK68CA 130453737 IC50 = 0.7 nM T97196 CDP9S1 130470501 IC50 = 10 nM T97196 C5U1XV 130470509 IC50 = 73 nM T97196 CLTQ15 130470516 IC50 = 63 nM T97196 CUO41K 130470684 IC50 = 0.6 nM T97196 CPC2A7 130470749 IC50 = 19 nM T97196 C7QI1J 131986481 IC50 = 5 nM T97196 CSWE45 134163712 IC50 = 360 nM T97196 CX0UR7 134694318 IC50 < 1.2 nM T97196 C9FUK2 135151360 IC50 = 17900 nM T97196 C81NTE 135980524 IC50 > 8000 nM T97196 C0AYN4 135980525 IC50 = 5800 nM T97196 CR4Z3O 137226388 IC50 > 40000 nM T97196 CTZA58 137628643 IC50 = 62 nM T97196 C0EY8G 138490470 IC50 = 22 nM T97196 CQ2M5F 138504490 IC50 = 1.8 nM T97196 CKDZ26 138504497 IC50 = 0.29 nM T97196 CH2D8T 145949518 IC50 > 28000 nM T97196 C9Q1TH 145950015 IC50 = 490 nM T97196 CK64FQ 145950570 IC50 = 23 nM T97196 C6JYA5 145950619 IC50 = 950 nM T97196 CPE7N3 145950719 IC50 = 130 nM T97196 CW6XJ2 145951187 IC50 = 160 nM T97196 CCOW60 145952011 IC50 = 240 nM T97196 CVR31U 145952361 IC50 = 6 nM T97196 C2WFH6 145953847 IC50 = 370 nM T97196 CTRQ36 145954357 IC50 = 100 nM T97196 CN7T2Q 145954771 IC50 = 8.6 nM T97196 CHR53Q 145957373 IC50 > 30000 nM T97196 C6R0OC 145957812 IC50 = 230 nM T97196 CA4C9J 145957925 IC50 = 8.2 nM T97196 C73CBD 145959061 IC50 = 230 nM T97196 C75LGW 145959260 IC50 = 1.7 nM T97196 CS13IP 145959347 IC50 = 1600 nM T97196 CDYO54 145959735 IC50 = 450 nM T97196 CS2KD5 145963991 IC50 = 3.9 nM T97196 CHRZ36 145964774 IC50 = 260 nM T97196 C6BQY4 145964941 IC50 = 140 nM T97196 C1I5GU 145964978 IC50 = 0.5 nM T97196 CCZ6K5 145966304 IC50 = 1.1 nM T97196 C9MB3A 145967469 IC50 = 0.9 nM T97196 CD71MG 145968213 IC50 = 35 nM T97196 C5K0LN 145969815 IC50 = 49 nM T97196 CZNQ73 145971262 IC50 = 3.9 nM T97196 C9R2VH 145971456 IC50 = 140 nM T97196 CVC90R 145971640 IC50 = 44 nM T97196 CRTG91 145973095 IC50 = 61 nM T97196 CN0EB3 145974305 IC50 = 27000 nM T97196 C07XEP 145977110 IC50 = 330 nM T97196 CGA83C 145981271 IC50 > 30000 nM T97196 C5R6BS 145987142 IC50 > 30000 nM T97196 C8X2IT 145996536 IC50 = 20 nM T97196 C9UF6S 155510524 IC50 = 3250 nM T97196 CH8J7L 155510809 Ki > 4000 nM T97196 C2MD1Q 155513187 IC50 > 10000 nM T97196 COM30P 155514391 Ki = 1400 nM T97196 CY1B4L 155517765 Ki = 400 nM T97196 CSPN68 155532569 Ki = 82 nM T97196 C23IEP 155536557 Ki > 10000 nM T97196 CG15CZ 155539194 IC50 = 132 nM T97196 C13HGT 155541849 IC50 = 70 nM T97196 CKIJ48 155543371 IC50 = 6000 nM T97196 CG7D9R 155543873 IC50 = 50 nM T97196 CBN29V 155544583 IC50 = 49 nM T97196 CW9F7M 155544669 IC50 > 30000 nM T97196 CHCS54 155546044 Ki = 1300 nM T97196 C6KXY5 155546286 IC50 = 3230 nM T97196 CPK82D 155546294 IC50 > 30000 nM T97196 CU2QO9 155547462 IC50 = 52 nM T97196 CY6F3D 155547951 IC50 = 908 nM T97196 CG8FO4 155548512 IC50 > 30000 nM T97196 C8JI1D 155550286 IC50 = 525 nM T97196 CQ5OD0 155550395 IC50 = 2 nM T97196 CAJ57R 155550406 IC50 = 606 nM T97196 CR8DO6 155550599 IC50 = 456 nM T97196 C5LTO0 155551695 IC50 = 418 nM T97196 CJL9K4 155552042 IC50 = 39 nM T97196 CJ75BO 155552100 IC50 = 0.8 nM T97196 CX6QO1 155552713 IC50 = 73 nM T97196 C2ZNL8 155552880 IC50 = 730 nM T97196 C09TOV 155553799 IC50 = 168 nM T97196 CHP3R7 155554099 IC50 > 30000 nM T97196 C0I4KF 155555078 IC50 = 373 nM T97196 CS8C4B 155555411 IC50 = 1130 nM T97196 C92NTS 155558433 IC50 = 45 nM T97196 CAV79P 155560264 IC50 > 30000 nM T97196 CO3R8Y 155560892 Ki = 105 nM T97196 C9UYA8 155561280 IC50 = 9700 nM T97196 CH9UY6 155562079 IC50 > 30000 nM T97196 CP52DQ 155562348 IC50 = 1840 nM T97196 CG9QR6 155563968 IC50 > 30000 nM T97196 CB7SJ5 155564720 IC50 = 137 nM T97196 CXKI62 155567017 IC50 = 571 nM T97196 C7KPT9 155567536 IC50 = 87 nM T97196 C8INK5 155568740 IC50 = 124 nM T97196 C1S8ZB 155568922 IC50 = 8 nM T97196 CQR7E9 155569091 IC50 > 30000 nM T97196 CE6P9C 155569571 Ki = 1350 nM T97196 D00MCG 16203946 IC50 > 10000 nM T97196 D00PXO 6605258 IC50 = 200 nM T97196 D01SXB 16203472 IC50 > 10000 nM T97196 D01ZMP 16203941 IC50 > 10000 nM T97196 D02SMG 16203943 IC50 > 10000 nM T97196 D02TSN 46244454 IC50 > 30000 nM T97196 D03DJC 16203354 IC50 > 100000 nM T97196 D03FTE 16204050 IC50 = 3200 nM T97196 D04DQF 16203469 IC50 > 10000 nM T97196 D05USL 5278396 IC50 < 2 nM T97196 D08WQW 16203714 IC50 > 10000 nM T97196 D09TJK 16203599 IC50 > 10000 nM T97196 D0F7ZK 16203255 IC50 > 10000 nM T97196 D0G0BJ 51000408 IC50 > 8000 nM T97196 D0K3VK 16203359 IC50 > 10000 nM T97196 D0KH8S 16203474 IC50 > 100000 nM T97196 D0O5BC 16204045 IC50 = 18000 nM T97196 D0PO9X 16204046 IC50 > 100000 nM T97196 D0QB9L 16204047 IC50 > 10000 nM T97196 D0R0TW 11964036 IC50 > 10000 nM T97196 D0S5SG 16203942 IC50 > 10000 nM T97196 D0T0BY 10039361 IC50 > 100000 nM T97196 D0W1ST 9860529 IC50 > 100000 nM T97196 D0X7TB 10017389 IC50 > 100000 nM T97196 D0Y3OO 11327430 IC50 > 100000 nM T97196 D0Z3CC 16204049 IC50 > 10000 nM T75984 D00TLN 2913 IC50 = 3.1 nM T75984 D01AZG 5073 Ki = 0.14 nM T75984 D01ZII 2726 Ki = 0.7 nM T75984 D05BMG 3007 Ki > 10000 nM T75984 D06ZUK 3696 Ki = 23 nM T75984 D08VRO 3822 Ki = 0.4 nM T75984 D08VYV 4168 IC50 = 13200 nM T75984 D0D1AL 3559 Ki = 4.2 nM T75984 D0F2PO 4828 Ki = 29500 nM T75984 D0K7WK 4595 Ki = 10000 nM T75984 D0M8VE 71360 IC50 = 9 nM T75984 D0PX8L 16351 Ki = 0.5888 nM T75984 D0R4OM 5566 Ki = 5.2 nM T75984 D0R6RO 4184 Ki = 1.1 nM T75984 D0TR5X 3386 IC50 > 100 nM T75984 D0U1OE 5452 IC50 = 18 nM T75984 D0U2OO 2477 Ki = 174 nM T75984 D0UA0I 28693 Ki = 0.3 nM T75984 D0V4QS 135398745 Ki = 12 nM T75984 D0WV3U 4893 IC50 = 42000 nM T75984 D0Z1RV 135398737 Ki = 1.8 nM T75984 D0ZS8P 2801 Ki = 8.3 nM T75984 D00POS 9931976 Ki = 168 nM T75984 D08CJK 1150 Ki = 50 nM T75984 D0C6QQ 60691 IC50 > 20000 nM T75984 D0Z2MB 6918107 Ki = 7800 nM T75984 D07YLK 4350931 Ki = 20 nM T75984 D00KZF 2419 Ki = 489.78 nM T75984 D00PXQ 60785 Ki = 0.26 nM T75984 D01RAE 133079 Ki > 1800 nM T75984 D01RCS 55752 IC50 = 2 nM T75984 D01WJZ 60820 Ki = 165 nM T75984 D02FNU 56971 IC50 = 10000 nM T75984 D03PJW 108029 Ki = 780 nM T75984 D03QMR 5685 Ki = 1000 nM T75984 D05MFO 71781 Ki = 12.5 nM T75984 D07MWD 44363475 IC50 = 0.9 nM T75984 D07ODD 132891 Ki = 377 nM T75984 D09DRG 9952420 IC50 > 1000 nM T75984 D09WHM 208917 Ki = 120 nM T75984 D0ES4S 183775 IC50 = 30 nM T75984 D0G1RT 132059 IC50 = 316.23 nM T75984 D0K8NW 5074 Ki = 0.26 nM T75984 D0K9JP 9928332 Ki = 144 nM T75984 D0L7BV 60547 Ki = 136 nM T75984 D0M7LV 5761 Ki = 2.5 nM T75984 D0M9GE 53389 IC50 > 50000 nM T75984 D0N1WM 122324 Ki = 4940 nM T75984 D0OS6O 60149 IC50 = 0.39 nM T75984 D0R9PL 9910257 Ki = 1006 nM T75984 D0V9HI 65845 IC50 = 3.4 nM T75984 D0X2TO 130918 Ki = 73 nM T75984 D0ZG9N 132337 Ki > 10000 nM T75984 C5JG6U 2689 IC50 = 6800 nM T75984 CZUI83 2769 Ki = 6.1 nM T75984 CR75OY 8423 Ki = 43300 nM T75984 C5H9CN 9287 Ki > 10000 nM T75984 CW3P5L 11297 Ki = 725 nM T75984 C4AL8P 11375 Ki > 300000 nM T75984 C3W0JR 11379 Ki = 79000 nM T75984 C93NZE 14641 Ki = 140 nM T75984 C7H2NQ 21138 IC50 = 7943.28 nM T75984 C1LOB9 31014 Ki = 1250 nM T75984 CSM9G2 31016 Ki = 16500 nM T75984 C5LAV6 31738 Ki > 10000 nM T75984 CU56WE 32593 Ki = 4 nM T75984 CTW48V 35758 IC50 = 2.6 nM T75984 C80INW 36431 IC50 = 740 nM T75984 CTB26S 52899 Ki > 10000 nM T75984 CBZ9E7 53263 Ki = 164.06 nM T75984 C4HB2O 55393 IC50 > 10000 nM T75984 CQ70DJ 55751 IC50 = 0.4 nM T75984 C27TKE 59750 IC50 > 10000 nM T75984 CR2EI3 60845 IC50 = 4817 nM T75984 CAF7T8 64622 Ki = 34 nM T75984 C9T4MY 68871 Ki = 37 nM T75984 CCL43X 70556 Ki > 10000 nM T75984 C05BAU 72038 Ki = 211 nM T75984 C13JOV 75994 Ki > 10000 nM T75984 CEHO46 91245 Ki = 1435 nM T75984 CB6G3Z 91536 Ki = 3500 nM T75984 C38YOB 91965 Ki = 558 nM T75984 CQ30NX 105432 Ki = 300 nM T75984 CF7BO0 119583 IC50 > 100000 nM T75984 CZ1KQ7 120580 Ki = 5 nM T75984 CZ9G2W 121264 Ki > 10000 nM T75984 CKR4N3 122065 Ki = 180 nM T75984 C8OQ0S 126060 Ki = 6.4 nM T75984 CC17JI 126589 Ki = 95 nM T75984 C9W8TH 127153 IC50 = 1179 nM T75984 C1PD0L 127887 Ki = 283 nM T75984 CN92EH 131396 Ki = 20 nM T75984 C5J8EX 131990 Ki = 281.84 nM T75984 C4PR2E 132564 IC50 = 14 nM T75984 CW8E1Q 133001 Ki = 1040 nM T75984 C9YA8O 134002 Ki = 1840 nM T75984 CKH16B 141047 Ki > 10000 nM T75984 CZHL23 146009 IC50 > 10000 nM T75984 CTUX03 147080 IC50 = 1000 nM T75984 CFV6Z2 150885 Ki = 180 nM T75984 C0ALO6 152215 Ki = 66.99 nM T75984 C93TIV 160463 Ki = 11500 nM T75984 CF3US2 169764 Ki = 1 nM T75984 CH7UQ2 174433 IC50 = 31.62 nM T75984 C3W4UK 182585 IC50 = 630.96 nM T75984 CU0BI8 184633 IC50 = 55.2 nM T75984 CX39NY 188249 Ki = 64.57 nM T75984 CAB98J 192260 Ki = 965 nM T75984 CA3T7R 192638 IC50 = 391 nM T75984 CD19AW 192639 IC50 = 770 nM T75984 C5A4GD 193381 Ki = 280 nM T75984 C87SEN 199116 Ki > 10000 nM T75984 CP76AJ 204291 Ki = 2525 nM T75984 CRZ9S5 212480 Ki = 415 nM T75984 CP7MR5 215369 Ki = 50 nM T75984 CNKZ62 215909 Ki = 70 nM T75984 CBKV12 226102 Ki = 3320 nM T75984 C2KIS9 240973 Ki = 3870 nM T75984 CA2S3F 244184 IC50 > 1000 nM T75984 C9O3CS 246532 IC50 > 1000 nM T75984 CX0M5S 316974 Ki > 150000 nM T75984 CV1B2K 332915 IC50 = 1670 nM T75984 CX1P9K 380265 Ki = 0.096 nM T75984 C6RHA8 448779 Ki = 4265.8 nM T75984 COMH91 542036 Ki = 218 nM T75984 CNT93E 542051 Ki = 69 nM T75984 CV9EI7 542053 Ki = 2200 nM T75984 CYZ25A 563919 Ki = 15.49 nM T75984 CIGF70 577725 Ki = 1580 nM T75984 CGIY90 688272 Ki > 1000 nM T75984 CU1R0C 762654 Ki > 10000 nM T75984 C9O5UM 765182 Ki > 10000 nM T75984 CXF82A 792043 Ki > 10000 nM T75984 C3TG9N 796570 Ki > 100000 nM T75984 C1BWS0 826664 Ki = 125 nM T75984 CE17JQ 854157 Ki = 5128.61 nM T75984 C8T9QW 899056 Ki > 10000 nM T75984 C8KX7N 899057 Ki > 10000 nM T75984 CK1HQ6 969502 IC50 = 5.623 nM T75984 CKIU74 1531644 Ki > 10000 nM T75984 CQ7G4J 2724440 Ki = 430 nM T75984 C4EX9F 2736460 Ki = 124 nM T75984 CNX3O2 2760448 Ki = 49000 nM T75984 CBGL54 3025750 Ki = 27.1 nM T75984 CS79YV 3028230 IC50 = 251.19 nM T75984 CW9Y2U 3036461 Ki = 142 nM T75984 C4TB0I 3036864 Ki = 13 nM T75984 CH8P2E 3046161 Ki = 3420 nM T75984 CUE91A 3055249 Ki = 897.43 nM T75984 C8UOQ7 3055329 Ki = 13.1 nM T75984 CFB6W2 3055343 Ki = 6.33 nM T75984 C3R8CQ 3055351 Ki = 9.78 nM T75984 C0BKW3 3055353 Ki = 37.6 nM T75984 CP8T5W 3055738 Ki = 1445.44 nM T75984 C04MWQ 3055752 Ki = 145.88 nM T75984 C58WXN 3061874 Ki = 51.05 nM T75984 CND8X6 3065055 IC50 = 1.9 nM T75984 CA9J3X 3065056 IC50 = 1.4 nM T75984 C5LB0E 3069816 IC50 = 125.89 nM T75984 C3WLF2 3070702 Ki = 13.9 nM T75984 CBHV93 3070706 Ki = 1.16 nM T75984 CAZ4J5 3070712 Ki = 41.3 nM T75984 CE8N7R 3081681 IC50 = 20 nM T75984 C5QF2D 3137663 Ki = 160 nM T75984 CTX1V4 3248000 Ki = 5.3 nM T75984 C2P5AH 3608822 Ki = 190 nM T75984 CQ0RN6 3699556 Ki = 64300 nM T75984 CCO5Y6 4092325 Ki = 570 nM T75984 C8C7VW 4742678 IC50 = 3200 nM T75984 CD3L7T 4742679 IC50 > 20000 nM T75984 C4NX5J 4742703 IC50 = 240 nM T75984 CQ94DZ 5274124 IC50 = 450 nM T75984 CGM63Y 6540428 Ki = 1.445 nM T75984 C4AV0Z 6603801 Ki = 35 nM T75984 CK69NC 6603907 Ki = 977.24 nM T75984 CSM9T8 6603950 IC50 = 0.48 nM T75984 CTPB95 6604720 IC50 = 199.53 nM T75984 CR48ZF 6604840 IC50 = 1393 nM T75984 CC6SM3 6618861 Ki = 43.55 nM T75984 CI0X2F 7059581 IC50 = 6.31 nM T75984 C1J3MK 9796025 Ki = 6309.57 nM T75984 CFC9Y5 9799318 Ki = 831.76 nM T75984 CG0UK3 9803482 Ki = 575.44 nM T75984 CR5XB1 9817779 Ki = 7.85 nM T75984 CR3KE7 9820675 Ki = 47 nM T75984 CC36YU 9820887 IC50 = 10 nM T75984 C9BI2T 9823904 IC50 = 22 nM T75984 CT26OQ 9826570 IC50 = 1.5 nM T75984 C32HEF 9842628 Ki = 2.13 nM T75984 CO8HB7 9844517 Ki = 75 nM T75984 CE3W4V 9845006 Ki = 112.2 nM T75984 CC24WR 9845261 IC50 = 28000 nM T75984 CCUB23 9845791 IC50 = 3.4 nM T75984 CD29OT 9854449 Ki = 395 nM T75984 C3EX7S 9862272 IC50 = 3.8 nM T75984 C8M5XK 9863333 Ki = 76 nM T75984 CVC3J6 9873473 IC50 = 8 nM T75984 C35LIA 9881324 IC50 = 17 nM T75984 CQ2BS0 9884087 Ki = 1.14 nM T75984 CTAC24 9885114 Ki = 1678 nM T75984 CL1W0B 9887186 Ki = 239.88 nM T75984 C2COG4 9888180 Ki = 89 nM T75984 C1CE9K 9889487 IC50 = 1.4 nM T75984 C6WY0D 9891901 Ki = 223 nM T75984 CL8B2Z 9894526 Ki = 722 nM T75984 CGX8H9 9894528 Ki = 1890 nM T75984 C6GZF9 9907305 Ki = 28.9 nM T75984 CO7BK6 9909648 Ki = 5.8 nM T75984 C9B3EA 9911844 Ki < 1000 nM T75984 CZBK50 9913230 IC50 = 1.1 nM T75984 CQ3YN1 9927016 IC50 = 1258.93 nM T75984 CZ4WE9 9927411 Ki = 6.2 nM T75984 CD50WC 9928073 Ki = 4.1 nM T75984 C4AB8C 9930706 Ki = 77 nM T75984 C2QB5N 9931837 IC50 = 1.5 nM T75984 CQ3AV4 9933918 Ki = 1360 nM T75984 CVH9B5 9956013 IC50 = 2.7 nM T75984 CHOJ30 9956365 Ki < 1000 nM T75984 C10EQY 9972693 Ki = 1148.15 nM T75984 CFSR80 9975973 IC50 = 205 nM T75984 CCZP34 9976750 IC50 = 398.11 nM T75984 CSM43E 9979063 IC50 = 16 nM T75984 C2LU8Z 9979258 IC50 = 6730 nM T75984 C24SWE 9981483 IC50 < 10 nM T75984 CHT1Y4 9992530 Ki > 10000 nM T75984 CXWA53 9993234 Ki = 10000 nM T75984 CFC14V 9993922 Ki = 0.62 nM T75984 C10DVM 9994615 Ki = 1078.95 nM T75984 CF0R6B 9995045 IC50 = 125.89 nM T75984 CX5Z9B 9995328 Ki = 1288.25 nM T75984 C9T1OG 9999042 Ki = 29 nM T75984 CJQ7H5 10002242 IC50 = 1.9 nM T75984 COI92B 10002473 IC50 = 20 nM T75984 CO4Q2N 10002491 IC50 = 140 nM T75984 CD9ZM6 10003405 IC50 = 5.7 nM T75984 C10SBA 10003806 IC50 = 18 nM T75984 CY53UZ 10003936 Ki = 94 nM T75984 CGVK68 10004551 IC50 = 1.6 nM T75984 CXT07W 10004580 IC50 = 49 nM T75984 C14PIV 10014625 Ki = 1729.82 nM T75984 C5ZJ4W 10015731 Ki > 5000 nM T75984 CHF2I4 10019227 Ki = 16 nM T75984 CP1E8D 10020976 Ki = 10 nM T75984 C7HU5C 10021562 IC50 = 204 nM T75984 C47SIL 10021763 Ki = 214 nM T75984 CMF0E8 10024423 IC50 = 3.5 nM T75984 CU2Q0B 10025027 IC50 = 0.78 nM T75984 C6J5MI 10025272 IC50 = 2.6 nM T75984 C4XQ5I 10025444 IC50 = 42 nM T75984 C1Z6GD 10025711 IC50 = 1170 nM T75984 CO9D5J 10025712 IC50 = 2370 nM T75984 C7ICY9 10026262 IC50 = 3.8 nM T75984 CJEA56 10026390 IC50 = 4.9 nM T75984 C1PFW3 10026395 IC50 = 1.6 nM T75984 CC8S0N 10026871 IC50 < 10 nM T75984 CP3B6I 10027633 IC50 = 89 nM T75984 COFD56 10035843 Ki > 10000 nM T75984 CVZ83J 10040938 Ki = 97.72 nM T75984 CAI92S 10042704 Ki = 1620 nM T75984 CG17SP 10043707 Ki = 16 nM T75984 C7U9JQ 10046480 IC50 = 2 nM T75984 CM14CY 10046952 IC50 = 5.1 nM T75984 C8U1BH 10047113 IC50 = 45 nM T75984 CPK3Z2 10047772 IC50 = 3.6 nM T75984 CRU83D 10047887 IC50 = 2.2 nM T75984 C5M0TX 10047977 IC50 = 91 nM T75984 CH64DF 10048445 IC50 = 2.8 nM T75984 C6N0FC 10048606 IC50 = 76 nM T75984 CI8O5M 10049666 IC50 = 5.2 nM T75984 CD7Y8O 10051181 IC50 = 241 nM T75984 C0Q4UK 10060720 Ki = 58 nM T75984 C1VPL9 10060979 Ki = 3097.42 nM T75984 C7XZ5C 10062773 Ki = 2805.43 nM T75984 CZL1K3 10063060 Ki = 984.01 nM T75984 CW6T5G 10066660 Ki = 6.5 nM T75984 C2U3ON 10067369 IC50 = 155 nM T75984 CZGI14 10069979 IC50 = 150 nM T75984 C24TYX 10070045 IC50 = 329 nM T75984 CG5B2A 10070289 IC50 = 111 nM T75984 CD0BT5 10071945 IC50 = 11 nM T75984 CAD78X 10073825 IC50 = 6 nM T75984 C2X7DL 10075243 IC50 = 2.9 nM T75984 C9HW3S 10085486 Ki = 7.7 nM T75984 CV04JN 10087023 Ki = 240 nM T75984 C3QFM9 10087566 Ki = 660 nM T75984 CS3AH6 10090259 Ki = 160 nM T75984 CKO26X 10090269 IC50 = 288 nM T75984 C7O8VH 10092041 IC50 = 220 nM T75984 C7L6QE 10093606 IC50 = 7.6 nM T75984 CY45PS 10093607 IC50 = 2.9 nM T75984 CZ15JC 10093723 IC50 = 2.3 nM T75984 CG70CM 10094790 IC50 = 8.5 nM T75984 CTO1Z3 10094822 IC50 = 1.9 nM T75984 CQ8WL5 10096660 IC50 = 7.9 nM T75984 CU9BX2 10097929 IC50 = 150 nM T75984 CB4W8T 10105889 IC50 = 680 nM T75984 CGE79A 10106586 Ki = 119.95 nM T75984 CX50IA 10108185 Ki = 1104.08 nM T75984 CYNF08 10108241 Ki = 1690.44 nM T75984 CE48KG 10108504 Ki = 1412.54 nM T75984 CT07DI 10220205 Ki = 230 nM T75984 C6K5ZM 10244251 IC50 = 81 nM T75984 CD8BW3 10245637 IC50 = 15 nM T75984 C0NT8I 10248163 IC50 = 417 nM T75984 C0E5SL 10248164 IC50 = 146 nM T75984 C0TXM6 10248523 Ki = 4.3 nM T75984 C94FIN 10250209 Ki = 274 nM T75984 C0UQ6P 10250792 IC50 = 209 nM T75984 CYG7W5 10252320 IC50 = 0.84 nM T75984 CZ6C4K 10254306 IC50 = 9.3 nM T75984 CS4W0E 10264302 Ki = 1348.96 nM T75984 C4SZ5U 10265917 Ki = 218.78 nM T75984 C98WGP 10266658 Ki = 50003.45 nM T75984 CTWJ70 10274894 Ki = 229.09 nM T75984 C3BEN4 10316605 IC50 = 104 nM T75984 CEK38I 10316830 Ki = 8.2 nM T75984 C80SEQ 10317012 IC50 = 40 nM T75984 C2N5XP 10319293 IC50 = 3.4 nM T75984 CIFD40 10319381 IC50 = 67 nM T75984 C2WRX3 10320252 IC50 = 122 nM T75984 CW5XO1 10320742 IC50 = 4.2 nM T75984 C4D2WS 10321139 IC50 = 170 nM T75984 C1AE8Y 10321140 IC50 = 41 nM T75984 C71YIK 10321160 IC50 = 1.3 nM T75984 CMW94R 10321674 IC50 = 20 nM T75984 CL2ZP4 10322234 IC50 = 4.5 nM T75984 C4N9QL 10322519 IC50 = 2.2 nM T75984 CCZO76 10323306 IC50 = 16 nM T75984 CN43AE 10335576 Ki = 512.86 nM T75984 CC08RY 10341964 IC50 = 5.8 nM T75984 CEI3H9 10342195 IC50 = 34 nM T75984 CH03FB 10342570 IC50 = 45 nM T75984 C8KX0R 10342773 IC50 = 391 nM T75984 C6DE9B 10343244 IC50 = 3.8 nM T75984 C7JO8R 10344071 IC50 = 143 nM T75984 CC5NR2 10344317 IC50 = 11 nM T75984 CS24DU 10353268 IC50 = 14 nM T75984 CX28TU 10354799 Ki = 7.87 nM T75984 C0AUN5 10356766 Ki > 10000 nM T75984 CSP30K 10356828 Ki = 2904.02 nM T75984 CX90VE 10360174 Ki = 44.67 nM T75984 CG9WL5 10361439 IC50 = 170 nM T75984 C38JVC 10361700 IC50 = 60 nM T75984 CKW5R3 10362229 Ki = 6.5 nM T75984 CR2HY8 10363225 IC50 = 26 nM T75984 CQS5V6 10364481 IC50 = 3 nM T75984 C2J1QR 10364835 IC50 = 1.6 nM T75984 CGQ4V3 10365032 IC50 = 0.73 nM T75984 C6DW2H 10365753 IC50 = 1.8 nM T75984 CC12QY 10378448 Ki = 5116.82 nM T75984 CE1XW6 10380005 IC50 = 199.53 nM T75984 CON6G8 10384067 IC50 = 147 nM T75984 CLY48W 10385977 IC50 = 330 nM T75984 CWY94C 10386748 Ki = 56.23 nM T75984 C7XP8H 10386866 IC50 = 36 nM T75984 CNQ5T7 10387365 IC50 = 1.8 nM T75984 CJ67LI 10387431 IC50 = 0.59 nM T75984 CHV45A 10387589 IC50 = 3.2 nM T75984 C2Z8WH 10387699 IC50 = 18 nM T75984 CGMB61 10389629 IC50 = 2.5 nM T75984 C1R7VZ 10401585 Ki = 19152 nM T75984 CXU73R 10401626 IC50 = 2511.89 nM T75984 CVQ9E8 10401691 IC50 = 398.11 nM T75984 CR6Y0F 10402195 Ki = 22387.21 nM T75984 C38WNT 10404819 Ki = 640 nM T75984 CDI85V 10406366 IC50 = 119 nM T75984 CY25MN 10407614 IC50 = 17 nM T75984 C7SDM0 10409070 IC50 = 3.1 nM T75984 CDKV19 10409784 IC50 = 1.1 nM T75984 C53AVT 10409893 IC50 = 7.9 nM T75984 C9R6GC 10411988 IC50 = 131 nM T75984 CWD56M 10421850 IC50 = 1584.89 nM T75984 C1YE2P 10425204 Ki = 53456.44 nM T75984 CD91FV 10426286 IC50 = 4.5 nM T75984 C5LJ8U 10427137 IC50 = 5.3 nM T75984 CN7HT1 10428802 Ki = 32 nM T75984 C1BAY5 10430858 IC50 = 63 nM T75984 CFR1U3 10431812 IC50 = 67 nM T75984 CNZ2C0 10432600 IC50 = 23 nM T75984 CT0HZ6 10432606 Ki = 51.29 nM T75984 CUM58D 10435274 IC50 = 38 nM T75984 C6O2MY 10452313 Ki = 655 nM T75984 CIL2T3 10452440 Ki = 12 nM T75984 CG5W7J 10452601 IC50 = 5.2 nM T75984 CLY07Z 10453320 IC50 = 2580 nM T75984 CA5C2U 10453356 IC50 = 5.5 nM T75984 CF09UT 10454460 IC50 = 53 nM T75984 CGHY35 10454774 IC50 = 2.3 nM T75984 C1Q2CU 10455211 IC50 = 0.9 nM T75984 C1IB2F 10455602 IC50 = 4.7 nM T75984 CGNZ49 10457262 IC50 = 1.3 nM T75984 CLW43J 10457974 IC50 = 3.7 nM T75984 CZ5Q6R 10467355 Ki = 7.84 nM T75984 CP4N9Y 10469060 Ki = 5128.61 nM T75984 CSC89H 10472257 Ki = 1760 nM T75984 CP56VK 10473320 IC50 = 33 nM T75984 C7GEB0 10474042 IC50 = 250 nM T75984 CTJR48 10474096 IC50 = 9140 nM T75984 CUE5J0 10475634 IC50 = 667 nM T75984 CCVN16 10476681 IC50 = 153 nM T75984 CKUZ19 10477439 IC50 = 3.2 nM T75984 C5W7DG 10478360 IC50 = 16 nM T75984 CLGR72 10478809 IC50 = 2.6 nM T75984 C51DVU 10482024 Ki = 27 nM T75984 C3P8FK 10493545 Ki > 5520 nM T75984 C9US6X 10497999 Ki = 230 nM T75984 CNU7J4 10498684 IC50 = 430 nM T75984 CN29IF 10500557 Ki = 42.66 nM T75984 CY8HR1 10500792 IC50 = 1200 nM T75984 C8N3XQ 10501072 IC50 = 85 nM T75984 C2EYI1 10501847 Ki = 38 nM T75984 CBT49U 10502415 IC50 = 2.3 nM T75984 CK5NO8 10502774 IC50 = 3 nM T75984 CKN3X1 10505718 IC50 = 16 nM T75984 CV2F0P 10505854 IC50 = 0.23 nM T75984 CJ2D6O 10522878 IC50 = 2720 nM T75984 C30TKY 10523786 IC50 = 2690 nM T75984 C3ZE8F 10524644 Ki = 114 nM T75984 CBQ4V1 10525589 IC50 = 1740 nM T75984 CAV9L4 10527245 IC50 = 3.4 nM T75984 CN0SA8 10528598 IC50 = 186 nM T75984 CZB50D 10537195 IC50 > 1000 nM T75984 C1A2YP 10548087 Ki = 71 nM T75984 C3K5RP 10549485 IC50 = 150 nM T75984 CCX26G 10550700 IC50 = 120 nM T75984 CH54UN 10550711 IC50 = 3.5 nM T75984 C9MPK1 10551250 IC50 = 1.6 nM T75984 CRC5S9 10551296 IC50 = 9.6 nM T75984 C27XLW 10551622 IC50 = 271 nM T75984 CL26QB 10553513 IC50 = 6.3 nM T75984 C6H2FI 10572440 IC50 = 439 nM T75984 C1UBL6 10572963 Ki = 1600 nM T75984 CB3K5S 10573307 IC50 = 2310 nM T75984 C1R2AS 10574164 IC50 = 2.2 nM T75984 CTOB12 10574209 IC50 = 134 nM T75984 C80HZB 10574309 IC50 = 5.8 nM T75984 CM7R6F 10574357 IC50 = 2.3 nM T75984 CD7Y8V 10574631 IC50 = 16 nM T75984 CYVW08 10575569 IC50 = 68 nM T75984 C6M9GL 10576037 IC50 > 20000 nM T75984 C7QR0I 10578206 IC50 = 12 nM T75984 C89NCX 10595767 IC50 = 588 nM T75984 CX0R6E 10596147 Ki = 961 nM T75984 C9K6IX 10597030 IC50 = 446 nM T75984 CI86FZ 10597953 IC50 = 90 nM T75984 CJT42R 10598597 IC50 = 2.3 nM T75984 CT8X6F 10599194 IC50 = 1.6 nM T75984 CZHX43 10600133 IC50 = 1.5 nM T75984 CA5C6E 10601553 IC50 = 45 nM T75984 C54LDF 10601561 IC50 = 6.8 nM T75984 CFC2L6 10601758 IC50 = 1.3 nM T75984 C2G4IR 10617200 Ki < 1000 nM T75984 CZB4V9 10619179 IC50 = 641 nM T75984 C56EVP 10620661 IC50 = 1270 nM T75984 C1WJK3 10621636 Ki = 180 nM T75984 C2DCY1 10622209 IC50 = 12 nM T75984 CRN41Q 10622408 IC50 = 1.6 nM T75984 CML9O4 10623136 IC50 = 196 nM T75984 CER8L0 10640982 Ki < 1000 nM T75984 C27CKV 10644772 Ki = 16.4 nM T75984 CLSG45 10645029 IC50 = 6 nM T75984 CQC82F 10645098 IC50 = 848 nM T75984 C9VU1L 10645711 IC50 = 3.2 nM T75984 C4EUS0 10646147 IC50 = 0.59 nM T75984 CZQY65 10646968 IC50 = 18 nM T75984 CEH17A 10647253 IC50 = 2 nM T75984 C0IKG5 10648292 IC50 = 2.3 nM T75984 CCK37J 10666322 IC50 = 569 nM T75984 CN40TJ 10668422 Ki < 1000 nM T75984 C0OKF3 10668966 IC50 = 1 nM T75984 C5BT6R 10669248 IC50 = 3300 nM T75984 CNS06L 10670032 IC50 = 2.4 nM T75984 C5EF0K 10672329 IC50 = 1110 nM T75984 C6IBF4 10672419 IC50 = 1.4 nM T75984 CO49AQ 10683127 Ki > 5000 nM T75984 C5H0WF 10689843 IC50 = 196 nM T75984 C1TN8V 10690470 IC50 > 1000 nM T75984 CH15KZ 10690544 Ki = 2180 nM T75984 CX9E7Q 10692544 IC50 = 492 nM T75984 CI8N9K 10692629 IC50 = 12 nM T75984 CG8YH7 10692833 IC50 = 3.9 nM T75984 CSZ4U9 10694912 IC50 = 105 nM T75984 C7ISC1 10695381 IC50 = 294 nM T75984 CP8A4L 10714760 IC50 > 10000 nM T75984 CQ7L4I 10715370 Ki = 514 nM T75984 C4NGW7 10715654 IC50 = 726 nM T75984 CJF35Z 10716365 IC50 = 349 nM T75984 CMB0Y6 10716503 IC50 = 3.9 nM T75984 CA5B3P 10717702 IC50 = 1.8 nM T75984 C65ZLE 10717711 IC50 = 18.9 nM T75984 CYK61A 10717745 IC50 = 1.8 nM T75984 C3RDH2 10717788 IC50 = 5.4 nM T75984 C6GQ7W 10717917 IC50 = 3.7 nM T75984 C4SH3J 10717919 IC50 = 1.4 nM T75984 CZ3A0O 10737314 Ki = 5.37 nM T75984 CHZY64 10739172 IC50 = 5 nM T75984 CPL4V2 10740625 IC50 = 43 nM T75984 C4RAC7 10740968 IC50 = 1710 nM T75984 C61BCK 10740969 IC50 = 841 nM T75984 CRQB19 10742244 IC50 = 51 nM T75984 CV1LT4 10744055 IC50 = 98.1 nM T75984 C59HIO 10744505 IC50 = 14 nM T75984 CO1JN2 10762097 IC50 = 8420 nM T75984 CW70SC 10763158 IC50 = 1560 nM T75984 CE6NL0 10763646 IC50 = 18 nM T75984 C62VHJ 10763976 IC50 = 428 nM T75984 C4IJQ1 10764716 IC50 = 1.7 nM T75984 CN9K8D 10764920 Ki = 348 nM T75984 C5FG6O 10765759 IC50 = 520 nM T75984 CZ42QL 10766150 IC50 = 3.8 nM T75984 C7XI0B 10767522 IC50 = 119 nM T75984 CN5DO0 10767648 IC50 = 26 nM T75984 C67LXV 10768199 IC50 = 30 nM T75984 C06HZP 10768266 IC50 = 15 nM T75984 C4SRZ8 10768312 IC50 = 142 nM T75984 CPTB50 10774576 Ki = 232 nM T75984 C5YUL9 10784211 Ki = 28 nM T75984 C3SWV9 10785714 Ki = 16.22 nM T75984 C2M9IZ 10785980 IC50 = 1900 nM T75984 C6HXP7 10786703 IC50 = 30 nM T75984 CRZ4X1 10786715 IC50 = 13 nM T75984 CNCQ18 10788417 IC50 = 8.9 nM T75984 CC68PW 10790896 IC50 = 53 nM T75984 C21MHD 10803229 Ki > 5520 nM T75984 C4VA1L 10805623 IC50 > 10000 nM T75984 CGX34B 10807793 Ki = 960 nM T75984 CO81ND 10809567 IC50 = 7 nM T75984 C1HW7E 10810014 Ki = 21 nM T75984 CNM42F 10811491 IC50 = 2.6 nM T75984 C75SKC 10811746 Ki = 104.71 nM T75984 C4T3FZ 10811983 IC50 = 2 nM T75984 C0L6MY 10812139 IC50 = 10 nM T75984 CIDB09 10812407 IC50 = 0.5 nM T75984 C3JV1Q 10812885 IC50 = 2040 nM T75984 C7Z8UD 10815075 IC50 = 126 nM T75984 C3JKY9 10822557 Ki = 227 nM T75984 C1E7LN 10830233 Ki = 180 nM T75984 C3DJ1I 10832067 IC50 = 8800 nM T75984 CLZH70 10833320 IC50 = 414 nM T75984 CS09YF 10833527 IC50 = 9.8 nM T75984 CG4X1R 10834268 Ki = 53.7 nM T75984 C3PD0J 10834424 IC50 = 503 nM T75984 C9PKC4 10834480 IC50 = 2.1 nM T75984 C8CEZ7 10836319 IC50 = 5.6 nM T75984 C03ZWR 10837325 IC50 = 1540 nM T75984 C1LMI8 10838359 IC50 = 580 nM T75984 C5Q4IJ 10862697 Ki = 64.57 nM T75984 CFY4V1 10862787 Ki = 97.72 nM T75984 CNEP25 10884517 Ki = 354.81 nM T75984 C67UIY 10884717 Ki = 537.03 nM T75984 C9S4ON 10891445 Ki = 3.1 nM T75984 C9C2FI 10895284 Ki = 97.72 nM T75984 CD4YL2 10896196 Ki < 1000 nM T75984 CEGJ41 10917174 Ki = 281.84 nM T75984 C7PWT9 10938620 Ki = 28.18 nM T75984 CA42MT 10939416 Ki = 812.83 nM T75984 C2MBP7 10949445 Ki = 39.81 nM T75984 C74SOA 10950559 Ki = 1380.38 nM T75984 C47MYE 10960943 Ki = 75.86 nM T75984 CJD58C 10971401 Ki = 114.82 nM T75984 CRS62E 11025847 Ki = 66.07 nM T75984 C0HA7O 11047374 Ki = 144.54 nM T75984 C80UIZ 11048252 Ki = 158.49 nM T75984 CONV96 11058267 Ki = 123.03 nM T75984 CD4BW6 11058564 Ki = 446.68 nM T75984 CI87XB 11059092 IC50 = 1.3 nM T75984 CZN25U 11059148 Ki = 45.71 nM T75984 C3AJ7L 11074351 Ki = 295 nM T75984 C15USQ 11101733 Ki = 524.81 nM T75984 C7OFQ4 11102049 Ki = 676.08 nM T75984 CCJ1U3 11112531 Ki = 1412.54 nM T75984 C5I0XL 11133795 Ki = 15.85 nM T75984 CS90QD 11145126 Ki = 758.58 nM T75984 C75WKP 11176199 IC50 = 20 nM T75984 CE60CJ 11197273 Ki = 517 nM T75984 C4SUZ1 11206672 Ki = 19.32 nM T75984 CC03FY 11287716 IC50 > 100 nM T75984 C9KZ5I 11301805 Ki = 74.9 nM T75984 CCF56T 11334373 Ki = 86.5 nM T75984 C4G5MW 11358431 Ki = 416 nM T75984 C3KE1Q 11361267 IC50 = 50 nM T75984 CV9D2U 11379561 Ki = 591.56 nM T75984 C0O3XY 11391950 Ki = 70.6 nM T75984 C7O8RQ 11460281 Ki = 4.55 nM T75984 C6W0IN 11495267 IC50 = 360 nM T75984 C9NYV7 11724078 Ki = 44.67 nM T75984 C18AKY 11724636 Ki = 180 nM T75984 CAF0J1 11725183 IC50 = 251.19 nM T75984 C2ML7T 11725312 IC50 = 1000 nM T75984 CV82QX 11729084 Ki = 131.83 nM T75984 CG72CS 11732538 Ki = 204.17 nM T75984 C69QEW 11735949 Ki = 60 nM T75984 C57IKL 11740526 Ki = 954.99 nM T75984 CXVS61 11741028 IC50 = 66 nM T75984 CT23IZ 11742071 IC50 = 0.082 nM T75984 C07CJI 11742411 IC50 = 2.9 nM T75984 CHE28U 11742887 IC50 = 0.82 nM T75984 CPT49Z 11744188 IC50 = 2 nM T75984 CABJ23 11745828 Ki = 146 nM T75984 C3YF0X 11754649 IC50 = 1.7 nM T75984 C4KNX5 11777180 IC50 = 3162.28 nM T75984 C2T3OV 11777228 IC50 = 794.33 nM T75984 CF2I9V 11777642 Ki = 957.19 nM T75984 CM9A7S 11777810 IC50 = 2511.89 nM T75984 CL4B3K 11778114 Ki = 2421.03 nM T75984 CYBH97 11779386 Ki = 25 nM T75984 C53BTN 11792324 Ki = 30 nM T75984 C9XJF2 11795179 Ki = 712 nM T75984 CR27BM 11795528 IC50 = 1.7 nM T75984 C3QK0F 11795529 IC50 = 5.5 nM T75984 CM9RP8 11796915 Ki = 277 nM T75984 CE5GA4 11797259 IC50 = 1070 nM T75984 CVP2X0 11798884 IC50 = 1060 nM T75984 C3PY7W 11811833 Ki = 371.54 nM T75984 CQV92N 11825614 Ki = 44.67 nM T75984 CW4BC2 11826723 Ki = 288.4 nM T75984 CJD8H3 12229248 Ki = 398.11 nM T75984 CR75NU 12262514 Ki = 19 nM T75984 CB8O1J 12312578 IC50 = 140 nM T75984 C8ANG1 12312582 IC50 = 110 nM T75984 CF4I5Y 12508857 Ki = 260 nM T75984 CL3S9X 12626561 Ki = 0.39 nM T75984 C28QEX 12765746 IC50 = 0.48 nM T75984 C2AXM7 12771208 Ki > 1000 nM T75984 CRF8I0 12771209 Ki > 1000 nM T75984 CH91YD 12772954 Ki = 1479.11 nM T75984 CNWD02 12852586 Ki = 67.6 nM T75984 CGDL21 12852637 Ki = 25.7 nM T75984 CN7C9J 12928517 IC50 = 723 nM T75984 C8C3HS 13015797 Ki = 2.1 nM T75984 CS7IM8 13154762 IC50 = 7.7 nM T75984 CK8IS6 13154764 IC50 = 4.9 nM T75984 CM6SW9 13154791 IC50 = 64 nM T75984 C5S8BW 13154792 IC50 = 21 nM T75984 COHL49 13200208 IC50 = 251.19 nM T75984 C2CY1U 13200213 IC50 = 63.1 nM T75984 C8FR3G 13200215 IC50 = 316.23 nM T75984 C4MVI8 13200217 IC50 = 158.49 nM T75984 CPQ30T 13200219 IC50 = 158.49 nM T75984 CUX4T0 13200221 IC50 = 398.11 nM T75984 CI4BZ0 13200223 IC50 = 199.53 nM T75984 CGR4W2 13200225 IC50 = 251.19 nM T75984 C2ZVJ0 13200227 IC50 = 398.11 nM T75984 CO1H8N 13200229 IC50 = 501.19 nM T75984 CLI76O 13200231 IC50 = 39.81 nM T75984 C9X2KY 13200236 IC50 = 251.19 nM T75984 C01WAN 13200239 IC50 = 630.96 nM T75984 CW0HY2 13200242 IC50 = 2511.89 nM T75984 CF8O1G 13200244 IC50 = 1584.89 nM T75984 C2MXQ8 13200246 IC50 = 158.49 nM T75984 C6L3BW 13200248 IC50 = 125.89 nM T75984 C0LR2N 13200250 IC50 = 251.19 nM T75984 CM7Y2R 13200252 IC50 = 158.49 nM T75984 C69EBI 13200254 IC50 = 501.19 nM T75984 C4T3CB 13200256 IC50 = 125.89 nM T75984 CT9PX7 13200258 IC50 = 501.19 nM T75984 CE7XC3 13200260 IC50 = 79.43 nM T75984 C16JUH 13200262 IC50 = 63.1 nM T75984 CMQ61Y 13200264 IC50 = 199.53 nM T75984 C2Z6MY 13200266 IC50 = 50.12 nM T75984 CIFP13 13200268 IC50 = 63.1 nM T75984 CL78OH 13200270 IC50 = 158.49 nM T75984 CT3DV2 13200272 IC50 = 79.43 nM T75984 CWCB64 13200274 IC50 = 2511.89 nM T75984 CH9W6L 13200279 IC50 = 158.49 nM T75984 CEB62Q 13200281 IC50 = 158.49 nM T75984 CTK61D 13200283 IC50 = 125.89 nM T75984 C0N7VC 13318472 Ki = 700 nM T75984 C2WFJ1 13356524 IC50 = 1756 nM T75984 CU8S2B 13437356 Ki > 10000 nM T75984 CWM47Z 13497176 Ki = 0.31 nM T75984 CNW08I 13547419 Ki = 25600 nM T75984 CHO4B1 13547420 Ki = 1930 nM T75984 CIR54H 13553507 Ki = 388 nM T75984 C1EL7Z 13580034 IC50 = 15444 nM T75984 C53FIX 13580045 IC50 = 390 nM T75984 C1PD2S 13599009 Ki = 76500 nM T75984 CBI41Y 13599017 Ki > 100000 nM T75984 C4U2VP 13599019 Ki = 93000 nM T75984 CMBD46 13646491 Ki = 602 nM T75984 CL1M5D 13673326 IC50 = 158.49 nM T75984 C68JVL 13772434 Ki = 173 nM T75984 CY02VP 13772438 Ki = 480 nM T75984 CR0GW4 13772450 Ki = 60 nM T75984 CVD25F 13781100 Ki = 94 nM T75984 CEF8R1 13781101 Ki = 8250 nM T75984 CV1W5Z 13900355 Ki = 9300 nM T75984 C0SGY4 13900359 Ki = 310 nM T75984 CWX4A8 13900384 Ki = 28 nM T75984 CJMU72 13900388 Ki = 55 nM T75984 CJGP87 13900392 Ki = 3.6 nM T75984 CB36WT 13900394 Ki = 23 nM T75984 CU78YH 13903117 Ki = 49 nM T75984 CNTO94 13903144 Ki = 7.4 nM T75984 CUAV93 13914131 IC50 = 3.9 nM T75984 CWE2L5 13914132 IC50 = 116 nM T75984 CM0A7C 13914133 IC50 = 43.4 nM T75984 CUTC50 13914137 IC50 = 70.9 nM T75984 CG6TW5 13914140 IC50 = 4.2 nM T75984 CN7V2Z 13914141 IC50 = 19.1 nM T75984 C5ZDJ7 13914143 IC50 = 6.7 nM T75984 C2H5XN 13914146 IC50 = 5.8 nM T75984 CHQA05 13914147 IC50 = 55.2 nM T75984 CLT7U9 13914149 IC50 = 5.7 nM T75984 CC7LF2 13914150 IC50 = 2.8 nM T75984 C36GOF 13914151 IC50 = 20.2 nM T75984 C6F5XO 14001256 IC50 = 199.53 nM T75984 CN26XL 14001258 IC50 = 100 nM T75984 CBVW95 14001260 IC50 = 3162.28 nM T75984 CX7T9K 14001262 IC50 = 3162.28 nM T75984 CMG0C2 14001264 IC50 = 3981.07 nM T75984 CENV53 14001265 IC50 = 10000 nM T75984 C61LOK 14001267 IC50 = 501.19 nM T75984 C5D9KT 14001269 IC50 = 199.53 nM T75984 C2NH5A 14001271 IC50 = 251.19 nM T75984 CS10KE 14001273 IC50 = 199.53 nM T75984 CQDF62 14001278 IC50 = 794.33 nM T75984 C9Z0DT 14001280 IC50 = 1000 nM T75984 CTJ74F 14001282 IC50 = 1258.93 nM T75984 CZ5RS6 14001284 IC50 = 501.19 nM T75984 C1SYH2 14001287 IC50 = 251.19 nM T75984 C4E0SQ 14001289 IC50 = 63.1 nM T75984 CY5K0R 14001291 IC50 = 794.33 nM T75984 C4MIL1 14001293 IC50 = 501.19 nM T75984 CQ5E7S 14011047 Ki = 7.1 nM T75984 CAM7Y3 14025825 Ki = 1400 nM T75984 CFBX75 14083209 Ki = 954.99 nM T75984 C3BEJ1 14083210 Ki = 1445.44 nM T75984 CHFN74 14083211 Ki = 707.95 nM T75984 CLJ94I 14083212 Ki = 1288.25 nM T75984 CJ6LH3 14083214 Ki = 6165.95 nM T75984 C7FQK5 14083215 Ki = 3467.37 nM T75984 C6RX9F 14083218 Ki = 3162.28 nM T75984 CP7BT4 14096630 IC50 = 1.1 nM T75984 CGN64J 14107776 IC50 = 1665 nM T75984 C24BRP 14107777 IC50 > 1000 nM T75984 CPE5H4 14107782 IC50 = 2650 nM T75984 CPCX96 14107786 IC50 = 3820 nM T75984 CJ25PF 14107790 IC50 = 1330 nM T75984 CMH38G 14107793 IC50 = 2120 nM T75984 CSE06V 14107796 IC50 = 210 nM T75984 COLB39 14107799 IC50 = 110 nM T75984 CRL9C1 14107802 IC50 = 1620 nM T75984 C2Q5FE 14107810 IC50 > 1000 nM T75984 CQ6CU2 14107812 IC50 = 1250 nM T75984 C71IOH 14107814 IC50 = 4220 nM T75984 C93AXV 14107816 IC50 = 1850 nM T75984 C7I3RX 14151595 IC50 = 178 nM T75984 CK2UF7 14151613 IC50 = 114 nM T75984 CB25MI 14151619 IC50 = 384 nM T75984 CH1F5R 14151633 IC50 = 920 nM T75984 CC5H0G 14151647 IC50 = 1100 nM T75984 C8YUJ3 14151657 IC50 = 1260 nM T75984 C6C9EM 14208318 IC50 = 30 nM T75984 CLE05X 14208320 IC50 = 18 nM T75984 CEN21T 14208321 IC50 = 570 nM T75984 CT7LI4 14208327 IC50 = 4.9 nM T75984 C92PIR 14208328 IC50 = 2.2 nM T75984 CI1JD4 14208331 IC50 = 11 nM T75984 CZ0N3V 14208332 IC50 > 1000 nM T75984 C47IHY 14208334 IC50 = 4800 nM T75984 CHT9M3 14208335 IC50 = 58000 nM T75984 CMZ9L0 14208336 IC50 = 5100 nM T75984 C59AZB 14208340 IC50 = 250 nM T75984 CK7B0H 14208341 IC50 = 310 nM T75984 CVKI82 14208342 IC50 = 6.5 nM T75984 CO9T3Z 14208343 IC50 = 4.3 nM T75984 CR6IF1 14208344 IC50 = 12 nM T75984 CV0LZ7 14208346 IC50 = 37 nM T75984 C8Z1XA 14208350 IC50 = 3.3 nM T75984 CIM15E 14208352 IC50 = 10 nM T75984 CEX8C3 14208353 IC50 = 4.8 nM T75984 CA10PX 14208355 IC50 = 4.8 nM T75984 C5YGT7 14208358 IC50 = 130 nM T75984 CDFP39 14208361 IC50 = 12 nM T75984 CWA4U2 14208364 IC50 = 3.3 nM T75984 CA3I9Y 14208365 IC50 = 5.6 nM T75984 CJMH71 14208367 IC50 = 22 nM T75984 CK57XG 14208369 IC50 = 7.5 nM T75984 CP8JH0 14208371 IC50 = 9.4 nM T75984 CHXM75 14208373 IC50 = 2.9 nM T75984 CS2D4R 14208374 IC50 = 3.4 nM T75984 C41ARP 14280585 IC50 = 390 nM T75984 CRK3F8 14280586 IC50 = 250 nM T75984 CM1X6A 14280588 IC50 = 3100 nM T75984 CWO9C8 14280593 IC50 = 8100 nM T75984 CU5DE6 14280599 IC50 > 20000 nM T75984 C8Q4VM 14280601 IC50 = 10 nM T75984 CJU53B 14280603 IC50 = 2700 nM T75984 CUZO58 14280605 IC50 = 10 nM T75984 CL48ZX 14450355 IC50 = 839 nM T75984 COC61N 14450361 IC50 = 86 nM T75984 CNEZ40 14450364 IC50 = 42 nM T75984 CSQ9P8 14450375 IC50 = 97 nM T75984 CI4O0M 14479835 Ki = 204 nM T75984 CDH6G0 14500867 IC50 = 1190 nM T75984 CQJP86 14580027 IC50 = 1 nM T75984 C5X3RF 14580031 IC50 = 6.3 nM T75984 CXW0T1 14580032 IC50 = 2.6 nM T75984 C0UMH3 14580033 IC50 = 0.2 nM T75984 CF82LY 14580034 IC50 = 0.3 nM T75984 C4H5LY 14580035 IC50 = 0.1 nM T75984 C17QDV 14580036 IC50 = 5 nM T75984 CYI1S9 14580038 IC50 = 7 nM T75984 C1EU7A 14580039 IC50 = 0.7 nM T75984 C48FAX 14580042 IC50 = 6.3 nM T75984 CKCW53 14623697 Ki = 198 nM T75984 C1O2JA 14726992 IC50 = 385 nM T75984 CE1I7Y 14727030 IC50 = 237 nM T75984 C07WUQ 14739622 Ki = 1550 nM T75984 C09YLK 14739623 Ki = 100 nM T75984 C1NH5V 14739624 Ki = 1040 nM T75984 C97MXQ 14739625 Ki = 140 nM T75984 CI4PF6 14739626 Ki = 280 nM T75984 C3H8TG 14739627 Ki = 635 nM T75984 CZFA63 14739628 Ki = 250 nM T75984 C7BSV6 14739640 Ki > 10000 nM T75984 C30DIW 14739643 Ki = 5200 nM T75984 CZVL61 14809027 Ki = 960 nM T75984 C8CKZ2 14816751 Ki = 21 nM T75984 CT6PY5 14894677 Ki > 10000 nM T75984 C5DO6I 14896472 IC50 > 20000 nM T75984 C5P2QX 14968310 Ki > 100000 nM T75984 CKXI45 14968311 Ki = 80 nM T75984 CT6ZD9 14968312 Ki = 34 nM T75984 CEL26N 14968313 Ki = 88 nM T75984 C94PMS 14968314 Ki = 32 nM T75984 CE9MG3 14968315 Ki = 70 nM T75984 CL1D2X 14968316 Ki = 95 nM T75984 C1Y2RI 14968317 Ki = 8 nM T75984 CDYQ49 14968318 Ki = 30 nM T75984 CLT34A 14968319 Ki = 5 nM T75984 C7PRK1 14968320 Ki = 325 nM T75984 CCR74L 14968321 Ki = 1000 nM T75984 CM3IL4 14968322 Ki = 600 nM T75984 CEK1U2 14973207 Ki = 354.81 nM T75984 C4L7WJ 14973208 Ki = 47.86 nM T75984 C4GY9E 14973209 Ki = 44.77 nM T75984 C3KM9T 14973210 Ki = 125.89 nM T75984 CR69IN 14973211 Ki = 557.19 nM T75984 C7GD4U 14973213 Ki = 16826.74 nM T75984 C9VQJ2 14973214 Ki = 3630.78 nM T75984 CNK50T 14973215 Ki = 4365.16 nM T75984 CB3W8C 14973216 Ki = 954.99 nM T75984 CWP28L 14973217 Ki = 10789.47 nM T75984 CFI1Q0 14975310 Ki = 688 nM T75984 CAX30B 14975317 Ki = 17.4 nM T75984 CV85FK 14975318 Ki = 15.9 nM T75984 C1W6NM 14975319 Ki = 35.9 nM T75984 C1KY7A 14975320 Ki = 9.3 nM T75984 C2M0TR 14978223 IC50 = 391 nM T75984 C9PB2V 14978224 IC50 = 119 nM T75984 C9UZ6Q 14978225 IC50 = 133 nM T75984 CK85WF 14978226 IC50 = 1170 nM T75984 CZ3RM5 14978227 IC50 = 932 nM T75984 CCE5S9 14978228 IC50 = 770 nM T75984 C9BTV5 14978229 IC50 = 205 nM T75984 C9FWE0 14978230 IC50 = 204 nM T75984 C52BPV 14978231 IC50 = 1340 nM T75984 C28LRH 14978232 IC50 = 2370 nM T75984 CD76OK 15006415 IC50 = 0.3 nM T75984 C1F9LG 15006416 IC50 = 4.4 nM T75984 CLRA60 15006441 IC50 = 3 nM T75984 C2UE9A 15006444 IC50 = 3.2 nM T75984 CDX9P6 15006448 IC50 = 2.7 nM T75984 C6UFS8 15006454 IC50 = 1.7 nM T75984 CPWM08 15006455 IC50 = 0.48 nM T75984 CVJ4D9 15006456 IC50 = 1.3 nM T75984 C5Y6UT 15006457 IC50 = 0.3 nM T75984 C0TV7N 15006458 IC50 = 1 nM T75984 C6VXM0 15006459 IC50 = 1 nM T75984 C1EAJ7 15006460 IC50 = 1 nM T75984 CI9K8Z 15006461 IC50 = 59 nM T75984 C7JKZ3 15006462 IC50 = 1.5 nM T75984 CJR84B 15006463 IC50 = 2.5 nM T75984 CR7K8F 15006464 IC50 = 0.24 nM T75984 C4K7RL 15006465 IC50 = 2.1 nM T75984 CU4I9R 15006467 IC50 = 4.4 nM T75984 C6F2KR 15006470 IC50 = 120 nM T75984 CP9D6A 15006472 IC50 = 25 nM T75984 CJ16HE 15011385 IC50 = 63 nM T75984 CN0KL5 15021875 Ki = 331.13 nM T75984 C5F7NM 15021876 Ki = 1.585 nM T75984 CE96NQ 15054215 IC50 = 249 nM T75984 CF2U3D 15061884 Ki = 2345 nM T75984 C48MNV 15121338 Ki = 14 nM T75984 C4QZU0 15121339 Ki = 19 nM T75984 CHLW54 15121340 Ki = 89 nM T75984 CNB0K1 15121341 Ki = 0.68 nM T75984 C3P4RZ 15121342 Ki = 9.6 nM T75984 CO6FT8 15121343 Ki = 37 nM T75984 CL95BR 15121344 Ki = 1.9 nM T75984 CTE54Y 15121345 Ki = 12 nM T75984 CW9LN2 15121346 Ki = 0.41 nM T75984 CYG4C7 15121347 Ki = 0.13 nM T75984 C0ZKG5 15121348 Ki = 1.1 nM T75984 CI3MP8 15121349 Ki = 1.3 nM T75984 CM3A5S 15121350 Ki = 3.2 nM T75984 CXF0M8 15121351 Ki = 1 nM T75984 C8SHM1 15121352 Ki = 4.4 nM T75984 CNM2J5 15124074 Ki = 355 nM T75984 CSY4X8 15124076 Ki = 267 nM T75984 CSU8G1 15128233 Ki = 825 nM T75984 C62RIN 15128236 Ki = 1030 nM T75984 CB9C1O 15128238 Ki > 10000 nM T75984 CS7QH6 15128241 Ki = 580 nM T75984 C9ADK4 15128244 Ki = 2460 nM T75984 C1SIX3 15183280 IC50 = 0.38 nM T75984 CTX2Z7 15233110 IC50 = 11000 nM T75984 C1QV8S 15284796 Ki = 26000 nM T75984 CKBD37 15542627 Ki = 891.25 nM T75984 C6A7SJ 15619872 Ki = 868.96 nM T75984 CQU06V 15619873 Ki = 4365.16 nM T75984 C05OLR 15619884 Ki = 286.42 nM T75984 C7V0BH 15646133 Ki = 0.8 nM T75984 C5V7FA 15646166 Ki = 1.87 nM T75984 CI9GO0 15646187 Ki = 4.25 nM T75984 CAX4S3 15646191 Ki = 6.11 nM T75984 CX8W7S 15646675 IC50 > 100 nM T75984 CT8QC2 15646681 IC50 = 45 nM T75984 CLP72C 15646682 IC50 = 11 nM T75984 C5CL3W 15646683 IC50 = 25 nM T75984 CADT05 15646684 IC50 > 100 nM T75984 CEP4I2 15646685 IC50 = 6 nM T75984 CA65BU 15646686 IC50 = 4.3 nM T75984 CU72XL 15646687 IC50 = 4 nM T75984 C8M2KZ 15646688 IC50 = 0.05 nM T75984 C0KOE7 15646689 IC50 = 16 nM T75984 CU4R3Z 15646690 IC50 > 100 nM T75984 CQ5M0Y 15646691 IC50 > 100 nM T75984 C29IOJ 15646692 IC50 = 23 nM T75984 C5WY1J 15646693 IC50 = 2.8 nM T75984 CG5S3X 15646694 IC50 = 72 nM T75984 CS0BX3 15646695 IC50 > 100 nM T75984 CU8Y5X 15646696 IC50 > 100 nM T75984 C6EPI7 15646697 IC50 = 4 nM T75984 C6QR8L 15646698 IC50 = 1.3 nM T75984 CV8SB5 15646699 IC50 = 6 nM T75984 CZ0N9S 15646709 IC50 = 27 nM T75984 CNZ07O 15646710 IC50 = 14 nM T75984 CEG46V 15646711 IC50 > 100 nM T75984 C3RV1K 15646712 IC50 > 100 nM T75984 CAO8Y2 15646713 IC50 = 100 nM T75984 CH4Z5S 15648963 IC50 = 0.53 nM T75984 C8ZK5G 15653098 IC50 = 40 nM T75984 C2YI0P 15653112 IC50 = 2.9 nM T75984 CKZ17A 15653113 IC50 = 2.8 nM T75984 C7PI1R 15653114 IC50 = 2.6 nM T75984 C6ZV9X 15653116 IC50 = 44 nM T75984 CJS70M 15653119 IC50 = 10 nM T75984 C4R8FN 15653120 IC50 = 5.6 nM T75984 CU06SQ 15653123 IC50 = 6.4 nM T75984 CJMO57 15653124 IC50 = 3.7 nM T75984 CHE4N3 15653125 IC50 = 3 nM T75984 CV45NJ 15653126 IC50 = 4 nM T75984 CE5N0O 15653127 IC50 = 9.9 nM T75984 C9L0GE 15653128 IC50 = 3.5 nM T75984 C3IY9C 15653129 IC50 = 26 nM T75984 C8F3GT 15653130 IC50 = 15 nM T75984 CY6QA4 15653131 IC50 = 11 nM T75984 C7DZS1 15654854 Ki = 124 nM T75984 C5C3AM 15654855 Ki = 48 nM T75984 C2HV6R 15654856 Ki = 124 nM T75984 CN04BU 15654858 Ki = 1870 nM T75984 C14OGI 15654859 Ki = 2900 nM T75984 CDR89S 15654860 Ki = 103 nM T75984 CS96IR 15654861 Ki = 7120 nM T75984 C3F4HY 15654862 Ki = 29 nM T75984 CNX75M 15654863 Ki = 2053 nM T75984 CD9J8C 15664993 Ki = 2300 nM T75984 CBS57T 15664994 Ki = 3700 nM T75984 CP17YH 15710725 IC50 = 2.1 nM T75984 CDK17W 15710726 IC50 = 11 nM T75984 CM4ZA7 15710727 IC50 = 7 nM T75984 CZ56EF 15710728 IC50 = 3 nM T75984 C2RK0N 15710729 IC50 = 18 nM T75984 CS62QM 15710730 IC50 = 25 nM T75984 CQ5EX0 15710731 IC50 = 4 nM T75984 CBV3J2 15710732 IC50 = 275 nM T75984 CUTG08 15710733 IC50 = 25 nM T75984 CI0S1D 15710734 IC50 = 200 nM T75984 CQ4H0L 15710735 IC50 = 32 nM T75984 C05IXG 15710736 IC50 = 2.3 nM T75984 CMC65S 15710737 IC50 = 0.4 nM T75984 CL8KM9 15710738 IC50 = 240 nM T75984 CL98VZ 15710739 IC50 = 540 nM T75984 CZW69A 15710740 IC50 = 1 nM T75984 CJG3S5 15710741 IC50 = 3.7 nM T75984 CR30OV 15710742 IC50 = 9.8 nM T75984 CFO7G8 15710743 IC50 = 5.1 nM T75984 CY2HD9 15710744 IC50 > 100 nM T75984 C6UBQ2 15710745 IC50 = 10 nM T75984 C0IY2G 15710746 IC50 = 10 nM T75984 C6US3O 15711850 Ki = 242 nM T75984 C5PO3N 15711869 Ki = 6360 nM T75984 C67CQH 15724475 Ki = 669 nM T75984 CTE25D 15724476 Ki = 1000 nM T75984 C8EK3G 15724477 Ki = 237 nM T75984 CEX14Y 15724478 Ki = 196 nM T75984 C97NCL 15724479 Ki = 1000 nM T75984 C8E7FD 15724480 Ki = 260 nM T75984 CM9B1P 15724483 Ki = 227 nM T75984 CKFZ62 15724484 Ki = 317 nM T75984 CHGY83 15724486 Ki = 409 nM T75984 C4YF6Z 15724487 Ki = 1000 nM T75984 C38LHI 15724488 Ki > 1000 nM T75984 C7WJ4U 15724490 Ki = 455 nM T75984 CH7U1M 15724491 Ki = 386 nM T75984 CTS31H 15724495 Ki = 256 nM T75984 CB3PV6 15724496 Ki > 100 nM T75984 CZV74S 15724497 Ki = 1000 nM T75984 C4O7HX 15724498 Ki > 100 nM T75984 CCH5S0 15724500 Ki = 137 nM T75984 C82PXH 15724502 Ki = 55.3 nM T75984 CXUV72 15724504 Ki = 669 nM T75984 COR32C 15724505 Ki = 110 nM T75984 C82GEF 15724507 Ki > 1000 nM T75984 CI6TS8 18377342 Ki < 1000 nM T75984 CHFJ09 18377388 Ki = 489.78 nM T75984 C5KB2J 18377409 Ki < 1000 nM T75984 CI91VX 18377415 Ki < 1000 nM T75984 CFQ7M8 18609309 IC50 = 320 nM T75984 CR4JL9 18609310 IC50 = 410 nM T75984 CH93CY 18649736 Ki = 2100 nM T75984 C23KVS 18649737 Ki = 300 nM T75984 C8Z2YT 18995769 Ki = 2.3 nM T75984 COHU81 18995773 Ki = 286 nM T75984 CZ1Q6B 18995777 Ki = 262 nM T75984 CE1C2J 19037250 IC50 = 1.5 nM T75984 CJ1SR2 19037269 IC50 = 0.95 nM T75984 C12WGX 19037273 IC50 = 1.1 nM T75984 CGY05I 19037281 IC50 = 120 nM T75984 C6K1YB 19037283 IC50 = 0.75 nM T75984 C4JXG1 19037286 IC50 = 1.5 nM T75984 CS97MG 19037289 IC50 = 8.9 nM T75984 C8KPF2 19037294 IC50 = 1.5 nM T75984 CH4Z1J 19774166 Ki = 50000 nM T75984 C4GB9F 19780145 Ki = 3000 nM T75984 C4HN6X 19780185 Ki = 2200 nM T75984 C4I2XO 20244201 IC50 = 5440 nM T75984 C94BPG 21460314 Ki = 125 nM T75984 C8EAU6 21768731 IC50 = 130 nM T75984 CA14GQ 22416530 IC50 > 1000 nM T75984 CW0V5M 22449331 Ki = 616.6 nM T75984 C3TRZ9 22826279 IC50 = 43 nM T75984 CZ7J4B 22857296 IC50 = 250 nM T75984 C89NDA 23277137 Ki = 84 nM T75984 CM6HF1 23277249 Ki = 3.1 nM T75984 C7MPO1 23786480 IC50 = 794.33 nM T75984 CA39DL 23844155 Ki = 1100 nM T75984 C1A9EF 23983765 Ki = 2.3 nM T75984 C6YE7C 24745966 Ki = 5.3 nM T75984 CCI50P 29010876 Ki = 54000 nM T75984 CFN0Q2 44265182 Ki = 7 nM T75984 C6FZ5D 44265202 Ki > 50000 nM T75984 C32VGM 44265214 Ki = 1530 nM T75984 CG76IH 44265221 Ki = 7550 nM T75984 CIH7T3 44265275 Ki = 76 nM T75984 CO0X7B 44265481 IC50 > 10000 nM T75984 CU04IV 44265483 IC50 = 146 nM T75984 CZI8A1 44267852 IC50 = 1258.93 nM T75984 C82RHM 44269026 Ki = 2.58 nM T75984 CS46GY 44269057 IC50 = 3 nM T75984 C1DX4N 44269058 IC50 = 280 nM T75984 CZ7UG8 44269068 Ki = 3 nM T75984 C97SDA 44269070 Ki = 33.4 nM T75984 C0L8KY 44269075 IC50 = 1220 nM T75984 C25NRU 44269092 IC50 = 120 nM T75984 CUS45A 44269094 IC50 = 2 nM T75984 C4PSK6 44269117 IC50 = 260 nM T75984 CIK9S1 44269120 IC50 = 430 nM T75984 C52KOG 44269131 IC50 = 520 nM T75984 CSIU30 44269132 IC50 = 610 nM T75984 CH8JO6 44269133 IC50 = 310 nM T75984 CH15BY 44269142 IC50 = 3 nM T75984 C8MRI0 44269143 IC50 = 4940 nM T75984 CVQ09T 44269145 IC50 = 32 nM T75984 C9MEF8 44269146 IC50 = 48 nM T75984 C1AT5B 44269148 IC50 = 54 nM T75984 CCV61I 44269165 IC50 = 540 nM T75984 CE0QG1 44271816 IC50 = 1.7 nM T75984 C3E5MW 44271822 IC50 = 1.6 nM T75984 CJI76W 44271870 IC50 = 2.7 nM T75984 C0IH5L 44274374 Ki > 1000 nM T75984 CZP13W 44274375 Ki > 1000 nM T75984 CZJE57 44274394 Ki > 1000 nM T75984 C3R1KH 44274590 Ki > 1000 nM T75984 C0KH4X 44282007 Ki = 54 nM T75984 CKTM89 44282450 Ki = 29 nM T75984 CLCS59 44283512 Ki > 10000 nM T75984 CVH2W7 44286416 IC50 = 0.69 nM T75984 CEPY31 44286775 IC50 = 4 nM T75984 CVNR05 44290349 Ki = 0.17 nM T75984 CLKY34 44296943 IC50 > 1000 nM T75984 C4I9KF 44297025 IC50 > 1000 nM T75984 C4A0EH 44298215 IC50 = 11.8 nM T75984 CQ89LH 44302841 Ki > 25000 nM T75984 CK9QN1 44312130 IC50 = 7943.28 nM T75984 CF2T6O 44312373 IC50 = 180 nM T75984 CIUB87 44316168 Ki = 71000 nM T75984 CI7Z2O 44316179 Ki = 50000 nM T75984 CM91QS 44317505 IC50 > 1000 nM T75984 CSV8L2 44317529 IC50 > 1000 nM T75984 C0TQ3U 44317536 IC50 > 1000 nM T75984 CNT8D3 44317537 IC50 > 1000 nM T75984 CU91NI 44317595 IC50 > 1000 nM T75984 CEO50M 44317596 IC50 > 1000 nM T75984 CA93MC 44319240 Ki = 691.83 nM T75984 C34FTE 44319435 Ki = 489.78 nM T75984 C5WB3L 44320050 Ki > 20000 nM T75984 CR7E3H 44320053 Ki > 20000 nM T75984 C8S7ZY 44320327 Ki > 20000 nM T75984 C7E4VR 44326342 IC50 = 12 nM T75984 CN2O1X 44326431 IC50 = 19 nM T75984 CCGT96 44331365 Ki = 1130 nM T75984 CU3Z7C 44331430 Ki = 125 nM T75984 C4JD8N 44331471 Ki = 1360 nM T75984 CG7RZ5 44331617 Ki = 716 nM T75984 CJW1P3 44331618 Ki = 82 nM T75984 CLQ9S5 44331619 Ki = 139 nM T75984 CK6BF0 44331666 Ki = 5360 nM T75984 CV5PX1 44331682 Ki = 3383 nM T75984 C9NR1G 44331683 Ki = 1035 nM T75984 C5GWJ6 44331703 Ki = 67 nM T75984 C8DTY2 44331704 Ki = 246 nM T75984 CXZK41 44331706 Ki = 165 nM T75984 C7UKT3 44331707 Ki = 14536 nM T75984 CG6H0L 44331726 Ki > 50000 nM T75984 C74YRV 44331727 Ki = 958 nM T75984 CU6G2T 44331743 Ki = 1070 nM T75984 C1N3SO 44331744 Ki = 139 nM T75984 C51ILW 44331758 Ki = 237 nM T75984 C3HW1U 44331759 Ki = 325 nM T75984 CG13OM 44331760 Ki > 50000 nM T75984 C76MOP 44331763 Ki = 146 nM T75984 CIT26J 44331775 Ki = 150 nM T75984 CP2LS3 44331776 Ki = 194 nM T75984 CCE1M0 44331777 Ki = 43 nM T75984 CR23BN 44331778 Ki = 107 nM T75984 C2EHY6 44346844 IC50 = 920 nM T75984 CMX45U 44348383 Ki = 0.3981 nM T75984 CHJ20E 44352359 Ki = 213.8 nM T75984 CAC4T8 44352376 Ki = 199.53 nM T75984 CH1PD3 44352408 Ki = 5000.35 nM T75984 C1U8FK 44363498 IC50 = 4.9 nM T75984 C9PJI4 44364724 Ki = 43.5 nM T75984 CTW3L2 44364825 Ki = 8.2 nM T75984 C9WC1P 44365113 IC50 > 1000 nM T75984 CDQ75B 44365114 Ki = 430 nM T75984 C8LB3Y 44365166 Ki = 170 nM T75984 C7B6EY 44365175 Ki = 430 nM T75984 C4ZM9C 44365177 Ki = 660 nM T75984 C2WY0V 44365298 IC50 > 1000 nM T75984 CDC2Q4 44365299 Ki = 160 nM T75984 CF8YS1 44372305 Ki > 1000 nM T75984 CT2BR5 44372581 Ki = 316.23 nM T75984 C0GX2T 44374544 Ki > 10000 nM T75984 C14WCF 44385319 IC50 = 147 nM T75984 CY02XS 44385451 Ki = 7.2 nM T75984 CXV9S0 44385452 Ki > 1000 nM T75984 C6YWM8 44385715 Ki = 13 nM T75984 C8BW9M 44385928 Ki > 1000 nM T75984 C2A1TN 44385979 Ki = 1700 nM T75984 CH3W7U 44385980 Ki = 1.3 nM T75984 CT8RZ5 44386356 IC50 = 2.6 nM T75984 C1YL3U 44386623 Ki = 0.09 nM T75984 C49YDI 44386833 Ki = 3.6 nM T75984 CO0H9E 44386836 Ki = 0.41 nM T75984 CK6C8V 44386883 Ki = 1 nM T75984 CO6L0A 44457584 Ki = 86 nM T75984 CS14UN 44457651 IC50 > 1000 nM T75984 CLFG23 44457652 Ki = 280 nM T75984 CSR4L5 44457668 Ki = 22 nM T75984 CC4DR7 44457669 Ki = 420 nM T75984 C4EQS8 44457680 Ki = 550 nM T75984 C2VJ1M 44457681 Ki = 99 nM T75984 CU16BT 44457682 Ki > 1000 nM T75984 C72ZAY 44457684 Ki > 1000 nM T75984 CXBJ25 44457685 Ki > 1000 nM T75984 CW60CO 44457756 Ki > 1000 nM T75984 C3JN6T 44457757 Ki > 1000 nM T75984 CK6ZB7 44457763 Ki > 1000 nM T75984 CLJD69 44457769 Ki = 400 nM T75984 CA1LC3 44457772 Ki > 1000 nM T75984 CIH50Z 44457774 Ki = 3300 nM T75984 CP73LK 44457795 Ki > 1000 nM T75984 CK17TR 44457796 Ki > 1000 nM T75984 CTSB98 44457797 Ki > 1000 nM T75984 CN5I3J 44460721 IC50 > 1000 nM T75984 C9IYB6 44460756 IC50 > 1000 nM T75984 C3B7MT 44460777 IC50 > 1000 nM T75984 C86HXK 44460799 IC50 > 1000 nM T75984 CX41DK 44461147 IC50 > 1000 nM T75984 C81TNO 45260709 IC50 = 10000 nM T75984 C20HND 45260721 IC50 = 251.19 nM T75984 CRV9G7 45263952 IC50 = 3.3 nM T75984 CA8KM6 45264562 IC50 = 1995.26 nM T75984 C86UAT 45264585 IC50 = 2511.89 nM T75984 C3CYV9 49799934 Ki = 3.7 nM T75984 C40SJM 52940491 Ki = 7 nM T75984 CM1VT5 52940568 IC50 = 13 nM T75984 CPJT83 52942993 IC50 = 12 nM T75984 C7YSJ0 52944126 Ki = 735 nM T75984 C91SBI 52944127 Ki = 3 nM T75984 C5GH8U 52944176 Ki = 10 nM T75984 CCPQ15 52944195 IC50 = 44 nM T75984 C12MFZ 52946610 Ki = 2400 nM T75984 CM29DS 52947773 Ki > 50000 nM T75984 C8IN6Z 52949018 Ki = 2.5 nM T75984 C4E9IQ 54580101 IC50 = 3.8 nM T75984 CF2A1J 54580952 Ki = 210 nM T75984 CCJI14 54581796 Ki = 29 nM T75984 CWVQ15 54583063 IC50 = 1.7 nM T75984 CX01ZC 54583776 IC50 = 15 nM T75984 C46WQA 54583789 Ki = 23.3 nM T75984 C8GL6W 54584896 Ki = 260 nM T75984 CS43YW 54585695 Ki = 8.5 nM T75984 CDC19B 54586952 IC50 = 6.1 nM T75984 CQ48AB 54587722 Ki = 252 nM T75984 C27WDI 57339832 Ki = 2250 nM T75984 CL0Q8T 57391435 Ki > 10000 nM T75984 CLZE69 71457959 IC50 = 11 nM T75984 C8A4HB 73352655 IC50 = 10 nM T75984 CF07BT 73354163 IC50 = 23 nM T75984 C78QXS 75105508 Ki = 4.3 nM T75984 CZ56GX 135423874 Ki = 3580 nM T75984 CT7XH1 135524906 IC50 = 28 nM T75984 CH96LU 135559170 Ki = 369 nM T75984 C2R4XT 136074292 Ki = 837 nM T75984 CMH8T1 136074293 Ki = 103 nM T75984 D00CGJ 13547422 Ki = 830 nM T75984 D00CRA 1574 Ki > 10000 nM T75984 D00FHZ 124007 IC50 > 10000 nM T75984 D00FUS 159755 Ki = 8130 nM T75984 D00PEU 4847 Ki = 0.3 nM T75984 D00QSV 152234 Ki = 7850 nM T75984 D00WEQ 62065 Ki = 0.79 nM T75984 D01APL 14987 IC50 = 160 nM T75984 D01KVG 9843179 Ki = 97.72 nM T75984 D01OGZ 71240 IC50 = 3.1 nM T75984 D01TOU 15139 Ki = 52 nM T75984 D01TSX 9840090 Ki = 9.9 nM T75984 D02AVN 1074765 Ki = 55600 nM T75984 D02ESW 107992 Ki > 1000 nM T75984 D02MVR 2761023 Ki = 203.7 nM T75984 D02OZB 70530 Ki > 1000 nM T75984 D02PLD 14479837 Ki = 277 nM T75984 D02SAF 2758473 Ki = 8430 nM T75984 D02TMK 1614 Ki = 2190 nM T75984 D02UWB 1809 Ki < 1000 nM T75984 D02XXA 12101308 IC50 > 1000 nM T75984 D02YFZ 2735875 Ki > 1000 nM T75984 D03CEZ 73484 IC50 = 270 nM T75984 D03NWV 83357 Ki = 774 nM T75984 D03PAH 410747 Ki = 3290 nM T75984 D03TDN 1342 Ki = 18 nM T75984 D04AQE 1833 Ki = 4.8 nM T75984 D04CTN 11074524 IC50 > 1000 nM T75984 D04VXP 2794808 IC50 = 377 nM T75984 D05EQG 5265 Ki = 0.45 nM T75984 D05QOF 14809026 Ki = 782 nM T75984 D05USH 17039492 Ki = 1100 nM T75984 D06OJI 13547424 Ki = 210 nM T75984 D06PKJ 62787 Ki = 465 nM T75984 D07LSC 77418 Ki > 1000 nM T75984 D07XTU 1229 Ki = 19 nM T75984 D08BCF 5011 Ki = 17 nM T75984 D08EFH 36906 Ki = 345 nM T75984 D08HOJ 34677 Ki = 11100 nM T75984 D08XYR 85875 Ki = 8 nM T75984 D08YJP 70529 Ki > 1000 nM T75984 D09JOE 13599004 Ki = 4710 nM T75984 D09OYA 2107 Ki = 125 nM T75984 D09YVA 44316216 Ki = 1200 nM T75984 D0A2BE 2780 Ki = 89 nM T75984 D0AJ3C 9819593 Ki = 415 nM T75984 D0B2GS 44372211 Ki = 8480 nM T75984 D0B3WX 5475158 IC50 = 2 nM T75984 D0C5XQ 1832 Ki = 15 nM T75984 D0C9TZ 44461148 IC50 > 1000 nM T75984 D0D2PL 22266820 Ki = 35000 nM T75984 D0D3OF 4738744 Ki = 2430 nM T75984 D0D3YN 1238 IC50 = 0.57 nM T75984 D0E2FY 10944016 Ki = 235 nM T75984 D0F6CD 5202 Ki = 6 nM T75984 D0F8TG 49381 Ki = 3.8 nM T75984 D0G0IQ 3802 Ki = 94 nM T75984 D0GI7S 3146743 IC50 > 1000 nM T75984 D0I4VT 44460502 Ki = 569 nM T75984 D0I9FI 205668 Ki = 4650 nM T75984 D0J1VB 10966027 IC50 = 141 nM T75984 D0J6JT 1355 Ki = 40 nM T75984 D0K5NZ 68848 Ki = 2 nM T75984 D0MU4A 5268 Ki = 113 nM T75984 D0N0LZ 10584082 Ki = 40 nM T75984 D0ND2Y 2760216 Ki = 419 nM T75984 D0O3GF 1220 Ki = 635 nM T75984 D0O9HS 415628 Ki > 1000 nM T75984 D0P0IX 16104 Ki = 1.778 nM T75984 D0P2HR 3510 Ki > 1000 nM T75984 D0R5QM 10354670 Ki = 2280 nM T75984 D0R7ZC 31721 Ki = 33600 nM T75984 D0S5ZY 44460743 Ki = 113 nM T75984 D0SP2J 10257 Ki = 380 nM T75984 D0T3IH 119146 Ki = 0.55 nM T75984 D0TH8D 22636319 Ki = 310 nM T75984 D0U1MN 10376185 Ki = 3120 nM T75984 D0U3GZ 98527 Ki = 34 nM T75984 D0V4RP 1346 Ki > 100 nM T75984 D0V5HV 4296 Ki = 31.1 nM T75984 D0V5SQ 68186 Ki = 2 nM T75984 D0W2YN 2760172 Ki = 70 nM T75984 D0X0PA 125379 Ki > 10000 nM T75984 D0X4RC 7096 Ki = 668 nM T75984 D0ZQ3Q 27402 Ki = 100 nM T85924 C7Y8VS 1318 IC50 = 185000 nM T85924 D0D7GL 10789 IC50 = 46800 nM T85924 D0H4YW 3611 IC50 = 24000 nM T89458 D0L4FS 5280961 Ki = 7000 nM T89458 D0Z0HH 3503 Ki = 20000 nM T89458 CYD71E 250016 IC50 = 11800 nM T89458 C3UE2I 1307491 IC50 = 180 nM T89458 C5T6UD 1385050 IC50 = 230 nM T89458 CAL0R8 1387075 IC50 = 50 nM T89458 CQJ9D2 1421264 IC50 = 270 nM T89458 CUM19E 1976692 IC50 = 1770 nM T89458 CTBV30 1977736 IC50 = 25 nM T89458 CC3FJ6 9996876 Ki = 98000 nM T89458 CHM36G 16033926 IC50 = 1500 nM T89458 CSZ12M 17017479 IC50 = 10 nM T89458 CO09IZ 28670291 IC50 > 100000 nM T89458 C8PLQ6 29105802 IC50 = 17 nM T89458 C08AQJ 42432904 IC50 > 100000 nM T89458 CX3J1L 44442294 Ki > 500000 nM T89458 CAH90M 44442299 Ki = 400000 nM T89458 CR51PF 44608046 IC50 = 4.9 nM T89458 C7GD2C 46830365 IC50 = 10900 nM T89458 CJUA36 52149799 IC50 = 510 nM T89458 C6RUX3 57412419 IC50 = 2000 nM T89458 CC9F3D 57413467 IC50 = 5000 nM T89458 C9QEL2 72547759 IC50 = 1 nM T89458 C7F3AZ 72548950 IC50 = 49 nM T89458 CK1R0M 72549874 IC50 = 7 nM T89458 C37WPK 72549875 IC50 = 35 nM T89458 C91QKT 72549876 IC50 = 4 nM T89458 C3LDR1 72550088 IC50 = 7 nM T89458 C3O4CK 72550310 IC50 = 5 nM T89458 C97JDB 72550752 IC50 = 150 nM T89458 CTWK21 72550753 IC50 = 10 nM T89458 C6J5MD 118191391 IC50 = 2 nM T89458 CM7F5P 118987010 IC50 = 267 nM T89458 C4VK7T 118987011 IC50 = 140 nM T89458 CEY03D 123183223 IC50 = 40 nM T89458 CN96KL 123249099 IC50 = 30 nM T89458 C6D8XT 123252892 IC50 = 8 nM T89458 C3N8QO 123482455 IC50 = 27 nM T89458 C3CZ2S 123753872 IC50 = 50 nM T89458 CGV12F 123899092 IC50 = 300 nM T89458 CDZ85L 123976747 IC50 = 20 nM T89458 C3R5OY 127029936 IC50 = 53 nM T89458 CD8IN2 127030110 IC50 = 33 nM T89458 CDTL03 127030174 IC50 = 80 nM T89458 CBJE45 127030175 IC50 = 100 nM T89458 CI0A4G 127030188 IC50 = 4400 nM T89458 C6AQ2R 127030417 IC50 = 200 nM T89458 CS10FZ 127030418 IC50 = 17 nM T89458 C5LMP6 127030492 IC50 = 4000 nM T89458 CE65PR 127031065 IC50 = 410 nM T89458 C7KO3Z 127031066 IC50 = 750 nM T89458 C3Y5MZ 127031374 IC50 = 1200 nM T89458 C4V7BO 127032848 IC50 = 1810 nM T89458 CE0QF7 127033761 IC50 > 10000 nM T89458 C9SDC1 127034087 IC50 > 10000 nM T89458 C37NJI 127034088 IC50 = 290 nM T89458 CJ0O1R 127034089 IC50 = 39 nM T89458 C8BI6U 127034090 IC50 = 110 nM T89458 CVC96B 127034091 IC50 = 180 nM T89458 C60QVK 127034096 IC50 = 230 nM T89458 CVM3H1 127034344 IC50 > 10000 nM T89458 CV7X6O 127034345 IC50 = 2400 nM T89458 CPKV38 127034346 IC50 = 1200 nM T89458 C4FS9U 127034354 IC50 = 9 nM T89458 CD7ZS8 127034355 IC50 = 60 nM T89458 CS5VD3 127034356 IC50 > 10000 nM T89458 CJ79OW 127034357 IC50 = 1900 nM T89458 C54FYT 127034358 IC50 = 470 nM T89458 CBX1O7 127034359 IC50 = 14 nM T89458 CR1WB5 127034364 IC50 = 120 nM T89458 C9BY8K 127034365 IC50 = 2300 nM T89458 C0H6JP 127034366 IC50 > 10000 nM T89458 CKN7B4 135186599 IC50 = 21800 nM T89458 C1Z4OQ 135187221 IC50 = 16000 nM T89458 CRVW26 135187266 IC50 = 28500 nM T89458 CY05WG 135187303 IC50 = 6500 nM T89458 CF50NU 135187499 IC50 = 4900 nM T89458 CJ45LW 135187505 IC50 = 20600 nM T89458 CU37QF 135187512 IC50 = 16900 nM T89458 CF8QE3 135187640 IC50 = 25800 nM T89458 CJT7X4 135187641 IC50 = 21000 nM T89458 C4V5MQ 135187645 IC50 = 28600 nM T89458 C2FK4X 135187669 IC50 = 16800 nM T89458 C8H2RO 135187678 IC50 = 11700 nM T89458 C3ICO4 135187683 IC50 = 12700 nM T89458 C9NOJ4 135187840 IC50 = 15600 nM T89458 CD06KP 135187841 IC50 = 21400 nM T89458 CKQ2T5 135187862 IC50 = 15100 nM T89458 CDPR31 136811094 IC50 = 450 nM T89458 C1Y7SP 137633968 IC50 = 32000000 nM T89458 CEF83K 137641243 Ki = 1200 nM T89458 C3ZL1N 137652693 IC50 = 65000 nM T89458 C3GSX9 137660299 Ki = 800 nM T89458 CA3W1K 155546221 IC50 = 10500 nM T89458 CWL5N6 155551084 IC50 = 4800 nM T89458 CJC5U6 155551654 IC50 = 6900 nM T89458 D0G3TK 5280863 IC50 = 4000 nM T89458 D0HD2G 4788 IC50 = 21400 nM T39664 CN5E3O 56969903 Ki = 24 nM T39664 CF45SA 118814313 Ki = 1541 nM T39664 CH84AT 122707109 Ki = 13 nM T39664 CIV02F 132991415 Ki = 7 nM T39664 CAOS95 132991416 Ki = 7 nM T39664 C92KTW 134132086 Ki = 17 nM T39664 CBD4E3 134135219 Ki = 132 nM T39664 CHJ93M 134136680 Ki = 50 nM T39664 C6X4AC 134138174 Ki = 135 nM T39664 CA6JW1 134139730 Ki = 21 nM T39664 CV94IW 134143316 Ki = 190 nM T39664 CO51QX 134144942 Ki = 47 nM T39664 C0XTH1 134145364 Ki = 9 nM T39664 CF0DX3 134147999 Ki = 190 nM T39664 CV0W1T 134151110 Ki = 86 nM T39664 C7M2XB 134151376 Ki = 97 nM T39664 CVBI19 134152354 Ki = 221 nM T39664 CP24SI 134154234 Ki = 63 nM T39664 CHFA70 134156979 Ki = 407 nM T39664 CFK1G0 134158354 Ki = 1.5 nM T39664 CK0B8Y 134158355 Ki = 42 nM T39664 CTI8A3 134158356 Ki = 58 nM T39664 CY1SG6 134158357 Ki = 6 nM T39664 CMW9T2 134158358 Ki = 12 nM T39664 CI2EW8 134158360 Ki = 9 nM T39664 C6SVY4 135567095 Ki = 64 nM T39664 C8NGI9 135567153 Ki = 7 nM T39664 CHQ5A1 135567209 Ki = 26 nM T39664 C94LEC 135567210 Ki = 11 nM T39664 C7PCS0 136042245 Ki = 245 nM T39664 CKC4Z8 136068369 Ki = 467 nM T39664 CUE0T5 137283267 Ki = 9 nM T39664 COHW89 137283360 Ki = 796 nM T39664 C1LMT5 137283363 Ki = 36 nM T39664 CQ4RS2 137292434 Ki = 405 nM T39664 C47JDH 137300714 Ki = 44 nM T39664 C2FOW1 137300715 Ki = 15 nM T39664 CO41ZN 145949471 Ki = 10 nM T39664 C7JQL3 145951052 Ki = 23 nM T39664 CNSK79 145951985 Ki = 2030 nM T39664 CFMG42 145955635 Ki = 6 nM T39664 C1HT3J 145956159 Ki = 686 nM T39664 CG62JF 145957633 Ki = 336 nM T39664 COUK32 145957805 Ki = 6 nM T39664 CJTH49 145960297 Ki = 34 nM T39664 CQAH97 145971773 Ki = 47 nM T39664 C27AQZ 145972421 Ki = 119 nM T71390 D08IWD 57363 IC50 < 0.1 nM T71390 D0A9YA 6918296 IC50 < 0.1 nM T71390 D02KRI 68741 IC50 = 0.18 nM T71390 D0J3CT 178077 IC50 = 11 nM T71390 D0S3XE 65986 IC50 = 55 nM T71390 D08JCL 11504627 IC50 = 256 nM T71390 D0Z9UB 166562 Ki = 1000 nM T71390 CL89PK 72899 Ki = 230 nM T71390 C3EP4O 81146 Ki = 40 nM T71390 CE7GN4 116469 Ki = 10000 nM T71390 CMXV58 130227 Ki = 0.4 nM T71390 CSD84A 132992 IC50 = 3.3 nM T71390 CF94PV 195410 IC50 = 2.1 nM T71390 CB7W8U 220047 Ki = 1000 nM T71390 CBY29G 260801 Ki = 30 nM T71390 CT41AK 348591 Ki = 10000 nM T71390 C20JCF 2735497 Ki = 10 nM T71390 C4QJ7Z 4777878 Ki = 310 nM T71390 CVF6K7 9805325 IC50 = 4 nM T71390 CS65UZ 9840531 IC50 = 3.2 nM T71390 C8G3MQ 9860236 Ki = 2000 nM T71390 CRO5V7 9882015 Ki = 260 nM T71390 CMU0C2 9888894 Ki = 85 nM T71390 CRYT14 9911625 IC50 = 0.07 nM T71390 C87KNG 9914880 IC50 = 0.5 nM T71390 CN0TU8 9915286 IC50 = 340 nM T71390 C3LF1G 9915313 IC50 = 1.8 nM T71390 CYPS97 9931818 IC50 = 9.8 nM T71390 CB9C5R 9977338 IC50 = 6.7 nM T71390 CA3DS4 9981612 IC50 > 1000 nM T71390 C3ZP7E 9981699 IC50 < 0.1 nM T71390 C05GWL 9983581 IC50 = 0.5 nM T71390 CKG54C 9996114 Ki = 60 nM T71390 C65EBK 9999375 IC50 = 0.88 nM T71390 C2YJD5 9999512 Ki = 100 nM T71390 C63ASZ 10000110 IC50 = 0.5 nM T71390 C02UNM 10003819 IC50 = 0.2 nM T71390 CBZ81M 10004171 IC50 = 7 nM T71390 C7BWP9 10006358 IC50 > 100000 nM T71390 C8T6ID 10017907 Ki = 35 nM T71390 CQ78VH 10022130 IC50 = 0.1 nM T71390 CY0KZ4 10022795 IC50 = 320 nM T71390 CLU2O3 10024326 IC50 = 0.58 nM T71390 C2Z8CJ 10028849 IC50 = 6 nM T71390 C7XKN2 10042260 Ki = 40 nM T71390 C2F3AX 10043081 IC50 = 0.3 nM T71390 C6M0EB 10045593 IC50 = 1.8 nM T71390 CJC2B8 10049013 IC50 = 0.2 nM T71390 C7LY9P 10064026 Ki = 10 nM T71390 CUJ3V9 10064949 IC50 = 340 nM T71390 CNBO36 10066927 IC50 = 0.08 nM T71390 CDX48K 10068571 Ki = 30 nM T71390 CC2O1D 10068872 IC50 = 0.6 nM T71390 CE1KY0 10069406 IC50 = 42 nM T71390 C58THN 10069491 Ki = 35 nM T71390 C97IAS 10073070 IC50 = 40 nM T71390 CTIV62 10074562 IC50 = 0.2 nM T71390 C1R9SW 10076629 IC50 = 930 nM T71390 CEFD67 10087827 IC50 = 6200000 nM T71390 CMR92F 10088855 Ki = 40 nM T71390 C2JFV1 10090787 Ki = 120 nM T71390 CE1A7B 10091434 IC50 = 8.1 nM T71390 CR80EN 10092299 IC50 = 5 nM T71390 CP0W5K 10092414 IC50 = 0.36 nM T71390 CAEL20 10092779 IC50 = 1.9 nM T71390 C70SHT 10093252 IC50 = 4.9 nM T71390 CSN6F7 10098124 IC50 = 0.16 nM T71390 C9IS3Z 10243712 Ki = 455 nM T71390 CK6EL5 10250238 Ki = 30 nM T71390 C2ZLN4 10250239 Ki = 38 nM T71390 C8MS3L 10250314 Ki = 35 nM T71390 C9WS6N 10250415 IC50 = 4.5 nM T71390 CW07NR 10251245 IC50 = 4.2 nM T71390 CBR9E2 10251725 IC50 = 60 nM T71390 C3FGC8 10254719 IC50 = 69 nM T71390 CTC01H 10254723 IC50 = 0.23 nM T71390 C2AK6N 10264096 Ki = 1000 nM T71390 C50LOX 10317887 IC50 = 5.7 nM T71390 CHJC79 10318954 IC50 = 1.3 nM T71390 CR9BY2 10318958 IC50 > 100 nM T71390 C7KIY2 10321847 IC50 = 12 nM T71390 CH47EK 10323494 IC50 = 0.4 nM T71390 CO5J0D 10339275 IC50 = 1.5 nM T71390 CIYU19 10340008 IC50 = 4.4 nM T71390 C4HEY8 10348441 IC50 = 0.5 nM T71390 CUY2B8 10361062 IC50 = 6.7 nM T71390 CNS54U 10361063 IC50 = 2.8 nM T71390 CC5Z7H 10362686 IC50 = 33 nM T71390 C8KG1C 10363135 IC50 = 0.2 nM T71390 CVM5I4 10365419 IC50 = 14 nM T71390 C5E4DI 10366549 IC50 = 2.1 nM T71390 CGD74S 10370345 IC50 = 0.12 nM T71390 CIRV78 10380223 Ki = 10000 nM T71390 C8ZS6T 10381969 Ki = 15 nM T71390 CW3AZ5 10386294 IC50 = 3.5 nM T71390 CO4XP8 10386420 IC50 > 100 nM T71390 C3L5QA 10387222 IC50 > 100 nM T71390 C6XQI3 10390536 IC50 = 0.09 nM T71390 CW60JR 10391141 IC50 = 0.13 nM T71390 CN0JS1 10406238 IC50 = 2.4 nM T71390 CJO4D3 10410339 IC50 = 29 nM T71390 C7TQA2 10411050 IC50 = 11 nM T71390 C2HVN8 10411536 IC50 = 0.04 nM T71390 CJV3F4 10413543 IC50 = 23 nM T71390 C2D9EA 10414585 IC50 = 0.2 nM T71390 CQY7J1 10422666 Ki = 2500 nM T71390 C73ABK 10428773 Ki = 20 nM T71390 CE92YM 10428890 Ki = 35 nM T71390 CB28ME 10429262 IC50 = 3.5 nM T71390 CK8L9B 10430264 IC50 = 1.4 nM T71390 CO8U9D 10436202 IC50 = 270 nM T71390 C12INV 10445491 Ki > 5000 nM T71390 C4WU5K 10450174 Ki = 10 nM T71390 CB2A3G 10452760 IC50 = 7.1 nM T71390 C7XG9K 10452763 IC50 = 2.3 nM T71390 C7HLC4 10452764 IC50 = 1.7 nM T71390 C42TKU 10453975 IC50 = 192 nM T71390 C2LG8W 10455880 IC50 = 71 nM T71390 C1TM7R 10469538 IC50 = 617 nM T71390 CWS2D8 10474701 IC50 = 50 nM T71390 CU5N9Y 10475240 Ki = 110 nM T71390 CWS15F 10476132 IC50 = 8.6 nM T71390 CGI56Y 10478160 IC50 = 0.4 nM T71390 C57HSJ 10481860 IC50 = 1.3 nM T71390 CQ30WC 10482892 IC50 = 0.09 nM T71390 C5N7PW 10500864 IC50 = 15 nM T71390 C51MLZ 10540212 IC50 = 3.5 nM T71390 CT3BX5 10588455 IC50 = 4200 nM T71390 C9EKA5 10730985 IC50 = 2.4 nM T71390 CY6D7I 10737132 IC50 = 5.5 nM T71390 CM28KN 10850018 IC50 = 2.9 nM T71390 CSWB97 10906263 IC50 = 6 nM T71390 C68QKD 10950495 IC50 = 130 nM T71390 C7VD0I 11004116 IC50 = 1200 nM T71390 CM53UN 11025709 IC50 = 210 nM T71390 C2BEY3 11101029 IC50 = 430 nM T71390 C4CSB9 11112715 IC50 = 1100 nM T71390 C5F3IC 11112792 IC50 = 410 nM T71390 CZ3YU8 11161937 IC50 = 4800 nM T71390 C5LX1F 11163404 IC50 = 295 nM T71390 CPY7N1 11173292 IC50 = 2100 nM T71390 CDIA87 11244952 IC50 = 553 nM T71390 C04TKS 11268166 IC50 = 119 nM T71390 C0SHF3 11303884 IC50 = 467 nM T71390 CE0V6Q 11381020 IC50 < 50 nM T71390 C31TGA 11486129 IC50 = 584 nM T71390 C5ANR8 11576377 IC50 = 113 nM T71390 CTM90A 11723281 Ki = 60 nM T71390 CAZ19Y 11724555 Ki = 30 nM T71390 COJ3Q0 11725152 Ki = 22 nM T71390 C5CAQ1 11726674 Ki = 85 nM T71390 CR5N7I 11755506 IC50 = 0.18 nM T71390 CGU4O8 11772392 IC50 = 9500 nM T71390 C1H7SB 11826346 IC50 = 3500 nM T71390 C96DPL 11855879 IC50 = 480 nM T71390 CC2GB0 14507074 Ki = 26 nM T71390 CL7NV9 15241375 IC50 > 1000 nM T71390 CIS9U1 15250735 IC50 = 1.4 nM T71390 C7CW2K 15347494 IC50 = 830 nM T71390 CPE7T0 18638060 Ki = 2200 nM T71390 C9V5RQ 19927034 Ki = 260 nM T71390 C2GAE5 21841475 IC50 = 570 nM T71390 COYL35 21841478 IC50 > 10000 nM T71390 C37XZW 21841488 IC50 > 10000 nM T71390 CU5Y3C 21841490 IC50 > 10000 nM T71390 CQEO41 21841508 IC50 > 10000 nM T71390 CM63SQ 22865060 IC50 = 870 nM T71390 CU6HP4 44264624 IC50 = 582 nM T71390 C9C4RK 44271130 IC50 > 100 nM T71390 CSV64F 44271133 IC50 = 1000 nM T71390 C4MD0O 44271147 IC50 > 1000 nM T71390 CCO08D 44271150 IC50 > 1000 nM T71390 CKYH52 44271172 IC50 > 100 nM T71390 C4AWP7 44271177 IC50 > 100 nM T71390 CIZ64F 44271186 IC50 > 100 nM T71390 C7MI6C 44271188 IC50 > 100 nM T71390 CT4XU9 44271189 IC50 > 1000 nM T71390 C6R0WD 44271195 IC50 = 18.4 nM T71390 C3JD5Z 44271203 IC50 > 100 nM T71390 CD1E0B 44271224 IC50 = 1000 nM T71390 C2NSM8 44271225 IC50 > 1000 nM T71390 C1FQ6O 44271232 IC50 > 1000 nM T71390 C8YEA5 44271245 IC50 > 1000 nM T71390 C45ZCB 44271246 IC50 > 1000 nM T71390 CE17GD 44271251 IC50 > 100 nM T71390 C0W1DK 44271252 IC50 > 100 nM T71390 C1D3AE 44271258 IC50 > 1000 nM T71390 C2VY7C 44271268 IC50 > 100 nM T71390 C2NWJ0 44271274 IC50 = 3.75 nM T71390 CM02PT 44271279 IC50 > 100 nM T71390 CU3P4D 44271283 IC50 > 1000 nM T71390 C7D2RT 44271314 IC50 > 1000 nM T71390 CBA70P 44271320 IC50 > 1000 nM T71390 CWI8M6 44274870 IC50 < 0.1 nM T71390 CK6FC9 44274900 IC50 = 41 nM T71390 CX6BV1 44274932 IC50 < 0.1 nM T71390 C8HK3W 44274947 IC50 = 25.2 nM T71390 CSN05C 44275112 IC50 = 10 nM T71390 C6JG8Z 44275130 Ki = 590 nM T71390 CWP7D4 44275145 IC50 = 154 nM T71390 CB7R1A 44275146 IC50 = 218 nM T71390 C8CI9L 44275160 Ki > 1000 nM T71390 CW15IV 44275169 Ki = 7 nM T71390 CMX5Q9 44275186 IC50 = 2.9 nM T71390 CL6W9P 44275190 IC50 = 212 nM T71390 CWXD82 44275204 IC50 = 0.2 nM T71390 C7HV2D 44275216 IC50 = 387 nM T71390 CASH41 44275218 IC50 = 0.4 nM T71390 CDW74N 44275219 IC50 = 1553 nM T71390 C73HPZ 44275234 IC50 = 0.2 nM T71390 CQI48U 44275235 IC50 = 1218 nM T71390 CXJ87U 44275236 IC50 = 381 nM T71390 CC6U2N 44275245 IC50 < 0.1 nM T71390 CQR65M 44275322 IC50 = 428 nM T71390 C0DQM8 44275323 IC50 = 1390 nM T71390 C15CZH 44275436 IC50 = 6300 nM T71390 CZ71SJ 44275446 Ki = 7 nM T71390 CDF20P 44275631 Ki = 35 nM T71390 CV0LC3 44277746 Ki > 2500 nM T71390 CRO7I0 44292736 IC50 = 2000 nM T71390 CSZ6E4 44292749 IC50 = 350 nM T71390 CYO73J 44292760 IC50 = 41 nM T71390 CCT13Z 44292770 IC50 = 870 nM T71390 C3EY8R 44292780 IC50 = 92 nM T71390 CF10PG 44293590 Ki = 30 nM T71390 CK2RJ9 44299652 IC50 = 180 nM T71390 CCED35 44314879 Ki = 0.8 nM T71390 CWNB98 44314892 Ki > 2500 nM T71390 C3TK6L 44314902 Ki = 1600 nM T71390 C2AC1R 44314907 Ki = 1600 nM T71390 CGI6N3 44314943 Ki = 1600 nM T71390 CLM49Y 44315410 IC50 = 0.2 nM T71390 CF7R9X 44315430 IC50 < 0.1 nM T71390 CJM7E9 44315474 IC50 < 0.1 nM T71390 CN58ZU 44315547 IC50 = 1.3 nM T71390 CTP9N0 44315618 IC50 = 4.5 nM T71390 C2DKW4 44315657 IC50 = 12 nM T71390 CI3E5Z 44315682 IC50 = 0.4 nM T71390 CO7ZU0 44315685 IC50 = 0.3 nM T71390 C9A0YC 44315700 IC50 = 1.7 nM T71390 CVD24Q 44315722 IC50 = 3000 nM T71390 CVAG48 44315739 IC50 = 6.7 nM T71390 CGXN06 44315740 IC50 = 1.7 nM T71390 C05YTO 44315755 IC50 = 5.7 nM T71390 CP49RD 44315756 IC50 = 29 nM T71390 CT0QB5 44315757 IC50 = 4.9 nM T71390 CZHB84 44315759 IC50 = 3.5 nM T71390 CM0KD2 44315819 IC50 = 0.1 nM T71390 CVYR32 44315864 IC50 < 0.1 nM T71390 C0DA9R 44315908 IC50 = 8.6 nM T71390 CV3X6A 44315969 IC50 = 4.2 nM T71390 C1WG6H 44315970 IC50 = 5 nM T71390 C2ORG3 44315992 IC50 = 40 nM T71390 CD27VS 44316012 IC50 = 1500 nM T71390 C9XR5K 44316040 IC50 = 42 nM T71390 C5C3VS 44316042 IC50 = 8.1 nM T71390 C8SKX0 44316063 IC50 = 1.8 nM T71390 C4UR6E 44316076 IC50 = 3.5 nM T71390 C2NG1P 44316077 IC50 = 2.3 nM T71390 C7NOY4 44322148 IC50 = 0.27 nM T71390 CJ4P8B 44322225 IC50 < 0.1 nM T71390 CXBF03 44329329 IC50 = 122 nM T71390 CJGD39 44338101 IC50 < 1 nM T71390 CM85RX 44338102 IC50 < 1 nM T71390 C6M9QA 44338152 IC50 = 0.1 nM T71390 C4IKG5 44338162 IC50 = 0.2 nM T71390 C3XU2H 44338163 IC50 = 0.2 nM T71390 C2V5CD 44338164 IC50 = 0.1 nM T71390 C4B0RA 44338187 IC50 = 0.2 nM T71390 C6T0PA 44338193 IC50 = 0.4 nM T71390 CBXO72 44338225 IC50 < 1 nM T71390 C9TSK2 44338226 IC50 < 1 nM T71390 CVD4I2 44338231 IC50 < 0.1 nM T71390 CIF8K9 44338238 IC50 = 10.2 nM T71390 C8REO3 44338254 IC50 = 0.2 nM T71390 CX9EB7 44338255 IC50 < 0.1 nM T71390 C1D9TE 44338287 IC50 = 25.2 nM T71390 CYMP02 44338289 IC50 = 1.6 nM T71390 CIQ50X 44338290 IC50 < 1 nM T71390 CQX4H3 44338298 IC50 = 1.4 nM T71390 C4ZTP0 44338299 IC50 < 1 nM T71390 CWY72O 44338303 IC50 = 2.2 nM T71390 CY87ER 44338307 IC50 < 0.1 nM T71390 C79VZY 44338311 Ki = 30 nM T71390 CQJ8F7 44338320 IC50 < 0.1 nM T71390 CFC71N 44338329 IC50 < 1 nM T71390 CD20EX 44338333 IC50 < 1 nM T71390 CO5ME9 44338343 IC50 = 7.9 nM T71390 CQM89S 44338379 IC50 = 24.6 nM T71390 CG4CX1 44338395 IC50 = 0.1 nM T71390 C3HTB0 44338396 IC50 = 0.3 nM T71390 C8Y1SR 44338430 IC50 < 0.1 nM T71390 C03SKL 44338440 IC50 < 0.1 nM T71390 CS84KM 44338457 IC50 < 1 nM T71390 C6G3QX 44338558 IC50 = 0.4 nM T71390 C53AIN 44338631 IC50 = 0.2 nM T71390 C56QUC 44338632 IC50 < 1 nM T71390 C3WMT4 44338668 IC50 < 1 nM T71390 CULP10 44338682 IC50 < 1 nM T71390 C8G9AH 44342447 IC50 = 830 nM T71390 CA2XO5 44342533 IC50 = 530 nM T71390 C5W4BM 44343165 IC50 = 260 nM T71390 CWPS98 44349957 IC50 = 5.4 nM T71390 C9ECO7 44349958 IC50 = 2120 nM T71390 C4WNL3 44350041 IC50 = 218 nM T71390 CMN9R2 44350093 IC50 = 147 nM T71390 CSO78L 44350227 IC50 = 428 nM T71390 CCO46E 44350228 IC50 = 330 nM T71390 C4YR2P 44350229 IC50 = 1300 nM T71390 C0E8OQ 44350239 IC50 = 580 nM T71390 CR6LZ1 44350246 IC50 = 443 nM T71390 C1RHZ6 44350258 IC50 = 125 nM T71390 C2SRP4 44350270 IC50 = 280 nM T71390 C0A6MU 44350284 IC50 = 1390 nM T71390 CDA84X 44350285 IC50 = 298 nM T71390 C0BV4E 44350286 IC50 = 2170 nM T71390 CE90TU 44350289 IC50 = 218 nM T71390 CMA2Z5 44350291 IC50 = 713 nM T71390 C97TQC 44350292 IC50 = 859 nM T71390 CCE5U6 44350293 IC50 = 1050 nM T71390 C7N9MR 44350326 IC50 = 280 nM T71390 CT1SC9 44350327 IC50 = 1100 nM T71390 CHQ9T5 44350334 IC50 = 1340 nM T71390 C3G7LK 44351555 IC50 > 10000 nM T71390 CH9XO4 44351556 IC50 = 1340 nM T71390 C7S8HU 44351573 IC50 = 550 nM T71390 C5GSO0 44351575 IC50 > 10000 nM T71390 CR83SY 44351601 IC50 > 10000 nM T71390 C9UA2Q 44351707 IC50 = 1400 nM T71390 CTS3J6 44351715 IC50 = 520 nM T71390 CGMQ98 44351716 IC50 > 10000 nM T71390 C7C5WX 44351747 IC50 > 10000 nM T71390 CA8M1B 44351848 IC50 = 52 nM T71390 CJM80V 44358932 IC50 = 9000 nM T71390 C6FR7H 44380957 IC50 = 12000 nM T71390 CP0VI9 44380958 IC50 = 15000 nM T71390 CKS13M 44381051 IC50 = 40000 nM T71390 CY4A9K 44381327 IC50 = 4000 nM T71390 CX1W8E 44381328 IC50 = 32000 nM T71390 CNUI84 44381333 IC50 > 100000 nM T71390 CY9SJ8 44383960 Ki = 320 nM T71390 CW5OQ7 44384007 Ki = 200 nM T71390 C2DR7X 44384008 Ki = 570 nM T71390 C8GU0Q 44384180 Ki = 790 nM T71390 CUH67A 44384235 Ki = 5000 nM T71390 C1S4JT 44384266 Ki = 52 nM T71390 CM4BC9 44384465 Ki = 7 nM T71390 CAWO81 44384470 Ki = 60 nM T71390 CC1D9W 44384471 Ki = 62 nM T71390 CV68YW 44384537 IC50 = 700 nM T71390 C0UYD4 44384538 Ki = 32 nM T71390 CO0M6G 44385025 Ki = 50 nM T71390 C6AMG5 44385110 Ki = 110 nM T71390 CB47GL 44385395 Ki = 170 nM T71390 C7U5PF 44391584 IC50 = 665 nM T71390 CLF8E2 44391595 IC50 = 372 nM T71390 COAB23 44391699 IC50 = 134 nM T71390 C9VUS0 44391700 IC50 = 166 nM T71390 CM4H1G 44391702 IC50 = 308 nM T71390 CK34ES 44391712 IC50 = 1200 nM T71390 CB69UH 44391721 IC50 = 1000 nM T71390 CIC71T 44391731 IC50 = 368 nM T71390 CV40UR 44391732 IC50 = 801 nM T71390 C79CYJ 44391758 IC50 = 1200 nM T71390 CZ7Q6H 44391760 IC50 = 255 nM T71390 CY4PH3 44391764 IC50 = 3300 nM T71390 C4Z5AS 46182749 IC50 = 13 nM T71390 CK4LV2 46182750 IC50 = 15 nM T71390 CBYI82 46905116 IC50 < 0.1 nM T71390 CUB32F 53319483 IC50 > 1000 nM T71390 CH37KT 53321999 Ki = 5000 nM T71390 CYO3H5 53322088 IC50 = 71 nM T71390 C8MDK2 66573464 IC50 = 26.5 nM T71390 C4NVH5 66574324 IC50 = 54.1 nM T71390 CX5N3W 66574325 IC50 = 22.1 nM T71390 CW7V1G 66574326 IC50 = 72.8 nM T71390 CMF67A 66574384 IC50 = 212.9 nM T71390 CTO13H 70689369 Ki = 220 nM T71390 CI6B9U 71454429 IC50 = 10000 nM T71390 C0SU7M 71461598 IC50 = 16000 nM T71390 C2IK3N 71716083 Ki = 110 nM T71390 CDW32B 71716701 IC50 = 83.9 nM T71390 CP8IY7 71717903 IC50 > 430 nM T71390 CE68DL 72708275 IC50 = 3.2 nM T71390 CJ3QN5 76309047 IC50 = 1.7 nM T71390 CQB36G 76316257 IC50 = 0.4 nM T71390 C49UDJ 76327181 IC50 = 0.3 nM T71390 CQ19BH 76327182 IC50 = 3.4 nM T71390 C9QZU8 118716738 IC50 = 50 nM T71390 CD01EI 118716739 IC50 = 8 nM T71390 CEZ9K2 127026663 IC50 = 83.8 nM T71390 CZ1K2O 127028927 IC50 = 15.6 nM T71390 C8CHF0 127028928 IC50 = 220.1 nM T71390 CL70XA 127029223 IC50 = 273.8 nM T71390 C2R7BN 127029225 IC50 = 157 nM T71390 C6FI9S 127034703 IC50 = 100000 nM T71390 CWQI76 127034923 IC50 = 98000000 nM T71390 CU4TE9 127035071 IC50 = 118000 nM T71390 CE7NL8 132531900 IC50 = 118800 nM T71390 CLS8M4 137631999 IC50 = 122000 nM T71390 C5EML0 137636913 IC50 = 35 nM T71390 CNT1U4 137640034 IC50 = 711 nM T71390 CS6M9W 137648691 IC50 = 29.3 nM T71390 C3I7JH 137654228 IC50 = 76.4 nM T71390 CX19MQ 155547708 IC50 = 480 nM T71390 D01AUS 11616925 IC50 = 119 nM T71390 D04AED 11509747 IC50 = 790 nM T71390 D04GZD 11695657 IC50 = 23 nM T71390 D04LXR 11515759 IC50 = 2800 nM T71390 D05XPT 11717189 IC50 = 27 nM T71390 D05ZPJ 6917653 IC50 = 1.9 nM T71390 D07BHS 11530398 IC50 = 45 nM T71390 D07BQG 11495248 IC50 = 5 nM T71390 D09KZA 10017278 IC50 = 579 nM T71390 D0M7OP 10106832 Ki > 1000 nM T71390 D0Q4GH 11501077 IC50 = 470 nM T71390 D0W6HB 10087225 Ki = 5 nM T71390 D0Z6BT 11702714 IC50 = 131 nM T15033 CDRB69 9885291 Ki = 770 nM T15033 C8FEG4 11857486 Ki = 8 nM T15033 CH3SY4 11857488 Ki = 7.8 nM T15033 C34JBI 11857680 Ki = 1100 nM T15033 CY8H4R 11858153 Ki = 560 nM T15033 C7I5WK 11964579 Ki = 28 nM T15033 C12JFO 11964663 Ki = 18 nM T15033 CA98QX 11964664 Ki = 4.7 nM T15033 C6JVN1 11965767 Ki = 3.9 nM T15033 CM0W9F 12073809 Ki = 29000 nM T15033 CU79WM 21035680 Ki = 8.1 nM T15033 C3Y0XZ 57692074 Ki = 30 nM T15033 CUZ3B8 58230405 Ki = 48 nM T15033 C9HBX4 58230406 Ki = 91 nM T15033 CXJW13 58230407 Ki = 51 nM T15033 CW4SR2 59799570 Ki = 100 nM T15033 C2GQ8H 66622526 Ki = 14 nM T15033 CFH79W 69440865 Ki = 10 nM T15033 C2C4RW 69441619 Ki = 44 nM T15033 CX7W5R 69442228 Ki = 280 nM T15033 CV86DX 71624890 Ki = 110 nM T15033 CKG96M 71624891 Ki = 91 nM T15033 CE0GS7 71625019 Ki = 43 nM T15033 C6B8IX 71625020 Ki = 8.3 nM T15033 CPD5U8 71625021 Ki = 220 nM T15033 CQ70HI 71625022 Ki = 320 nM T15033 CHR84P 71625024 Ki = 600 nM T15033 CC0O7K 71625143 Ki = 220 nM T15033 CR4C3X 71625144 Ki = 640 nM T15033 CD0ZE4 71625145 Ki = 1200 nM T15033 CDC34R 71625146 Ki = 190 nM T15033 CK4J5A 71625271 Ki = 4 nM T15033 C0U6DF 71625272 Ki = 23 nM T15033 C0A6VG 71625273 Ki = 70 nM T15033 CM6KB1 71625274 Ki = 120 nM T15033 CXHS27 71625275 Ki = 99 nM T15033 C43XWU 71625276 Ki = 32 nM T15033 C3EG4B 71625389 Ki = 47 nM T15033 CY2RQ6 71625390 Ki = 1200 nM T15033 CP4QS0 71625391 Ki = 71 nM T15033 C6CW4Y 71625392 Ki = 360 nM T15033 CN83DJ 71625501 Ki = 670 nM T15033 C7S0CI 71625502 Ki = 900 nM T15033 CQ2Z3N 71625503 Ki = 18 nM T15033 C9N4FO 71625504 Ki = 110 nM T15033 C7Q2FV 71625505 Ki = 13 nM T15033 C2GKN5 71625506 Ki = 102 nM T15033 CP9E7K 71625625 Ki = 42 nM T15033 C1N4GD 71716556 Ki = 6.2 nM T15033 CA89MZ 71718998 Ki = 5.8 nM T15033 C7RUD1 71720196 Ki = 21 nM T15033 C6ENV5 100951623 EC50 > 10000 nM T90553 D0E3TC 44259 IC50 = 0.438 nM T90553 D0O6ZO 9952773 IC50 > 10000 nM T90553 CWM18I 11406175 IC50 > 10000 nM T90553 C1WXC5 11417488 IC50 = 1508 nM T90553 CTG83F 11539329 Ki > 6700 nM T90553 CACS26 11561968 Ki > 2000 nM T90553 CMIL86 11590363 Ki > 6700 nM T90553 C9T6SC 11640926 Ki > 6700 nM T90553 CU0E8O 11690457 Ki > 5000 nM T90553 CFPW41 16007116 Ki > 6700 nM T90553 C7YG1N 24759534 IC50 = 1 nM T90553 CX1HL8 25032704 Ki > 6670 nM T90553 CA51SY 25141108 IC50 < 0.25 nM T90553 C87WKU 25205097 IC50 = 70 nM T90553 CETQ79 44427518 IC50 = 3650 nM T90553 COPG94 44427519 IC50 > 10000 nM T90553 CLI16E 44465026 IC50 = 20 nM T90553 CY3HW5 46224684 IC50 = 210 nM T90553 CLS29B 46872626 IC50 > 10000 nM T90553 C2XTV7 59603828 IC50 = 24 nM T90553 CXJ63M 59603829 IC50 = 6 nM T90553 CQEU96 59603842 IC50 <= 0.5 nM T90553 C09FVB 59603906 IC50 = 1.3 nM T90553 C1M4WZ 59603929 IC50 = 99 nM T90553 CW4QG3 59603981 IC50 = 13 nM T90553 CV63UL 67240318 IC50 > 10000 nM T90553 C9E1NC 68776463 IC50 = 1 nM T90553 CZV54F 68777548 IC50 = 129 nM T90553 C9E8XL 68778264 IC50 = 9 nM T90553 CLR0X7 68779790 IC50 = 43 nM T90553 C5DGR9 69036886 IC50 = 1.2 nM T90553 CPA02V 70841494 IC50 = 5 nM T90553 C1DEQ6 70942743 IC50 = 37 nM T90553 CKT60L 71455860 Ki = 4830 nM T90553 CJ2T9E 76332983 IC50 > 10000 nM T90553 C1HW4B 89735655 IC50 = 5 nM T90553 CH9BP3 127021001 IC50 = 61 nM T90553 C0LY3A 134129875 IC50 = 2100 nM T90553 C6K1TJ 134130033 IC50 = 82 nM T90553 CHV40L 134130103 IC50 = 850 nM T90553 C1Q2AZ 134130107 IC50 = 2564 nM T90553 C7OK6L 134130144 IC50 = 2800 nM T90553 CCW4O0 134130175 IC50 = 226 nM T90553 CDP7Q0 134130181 IC50 = 304 nM T90553 CT5RL6 134130320 IC50 = 60 nM T90553 C12UXV 134130374 IC50 > 30000 nM T90553 C0GRK2 134130397 IC50 = 10 nM T90553 CHQB27 134130448 IC50 = 1524 nM T90553 C18VDQ 134130540 IC50 = 738 nM T90553 CNU0C2 134130690 IC50 = 10 nM T90553 CW3LI4 134130692 IC50 = 80 nM T90553 COX75D 134130730 IC50 = 2800 nM T90553 CJ86AV 134130841 IC50 = 627 nM T90553 CR4TU9 134130878 IC50 = 3000 nM T90553 CM79UL 134130892 IC50 > 30000 nM T90553 C3PR8Q 134130943 IC50 = 14 nM T90553 C08NTZ 134130961 IC50 = 1300 nM T90553 CX51VI 134131112 IC50 = 80 nM T90553 C24LZQ 134131373 IC50 = 1644 nM T90553 C9MXN1 134131388 IC50 = 120 nM T90553 CLG07B 134131413 IC50 = 12770 nM T90553 C02IUK 134131474 IC50 = 4300 nM T90553 CIA49M 134131483 IC50 = 27 nM T90553 CLY29G 134131496 IC50 = 346 nM T90553 CHJ0V1 134131530 IC50 = 1800 nM T90553 CNO5B2 134131560 IC50 = 19 nM T90553 C7YJ0G 155510540 IC50 = 10 nM T90553 C2MD1Q 155513187 IC50 > 10000 nM T90553 C39XGN 155544039 IC50 = 38 nM T90553 CEQO14 155544899 IC50 = 2 nM T90553 CUL01O 155551158 IC50 = 74 nM T90553 CWPX61 155554602 IC50 = 15 nM T90553 CY9N1O 155555954 IC50 = 2.4 nM T90553 C03IWC 155558700 IC50 = 3 nM T90553 CP8HY3 155559157 IC50 = 130 nM T90553 CIGR98 155560320 IC50 = 10 nM T90553 CWCZ68 155562819 IC50 = 9 nM T90553 CI8LZ2 155564791 IC50 = 15 nM T90553 C9OI7A 155568523 IC50 = 22 nM T90553 D00ERW 44444843 Ki > 6667 nM T90553 D00HVA 11624601 Ki > 6700 nM T90553 D03BJF 44465558 IC50 = 12 nM T90553 D0Q3NG 11715520 Ki > 6700 nM T90553 D0S7IE 11658882 Ki > 6700 nM T34099 D0Y7PG 4659569 IC50 = 640 nM T34099 CSHM20 73201 Ki = 345000 nM T34099 CPZ4O3 257767 IC50 = 2750 nM T34099 CBA61G 282274 IC50 = 1800 nM T34099 CTD9M6 427880 IC50 = 14400 nM T34099 CY63GZ 636530 Ki = 21000 nM T34099 CYO4C2 641785 Ki = 377000 nM T34099 COK25V 5289155 EC50 = 4500 nM T34099 C13KBC 5730111 IC50 = 2940 nM T34099 C7UVE8 6420188 Ki > 500000 nM T34099 C82ILF 6483648 Ki = 25000 nM T34099 C2RWJ3 6857723 Ki = 5800 nM T34099 CEMJ16 7188277 Ki = 7000 nM T34099 C47BJO 11343373 Ki = 12000 nM T34099 CL19OM 11635300 Ki = 1500 nM T34099 C39WCF 11974466 Ki = 61400 nM T34099 CQ8G6R 11974564 Ki = 113300 nM T34099 CHT2K6 11974565 Ki = 51000 nM T34099 CMQ8V2 11974566 Ki = 115000 nM T34099 CG2QC0 11974567 Ki = 9400 nM T34099 CUT79K 11974634 Ki > 500000 nM T34099 CW78CO 11974635 Ki = 5300 nM T34099 CK0X7G 11974636 Ki = 40700 nM T34099 CH67YL 11974637 Ki = 6800 nM T34099 C3JPI8 11974638 Ki = 33000 nM T34099 C5UZK8 11974730 Ki = 18600 nM T34099 CX69GQ 11974732 Ki = 7500 nM T34099 CL4MI1 11974733 Ki = 138000 nM T34099 C5YPR9 11974734 Ki = 41300 nM T34099 CYXZ51 11974839 Ki = 47400 nM T34099 C3BRG8 11974840 Ki = 43700 nM T34099 C30BZE 11974841 Ki = 28600 nM T34099 CO0RN6 11974842 Ki = 193000 nM T34099 C8DR5Q 11974843 Ki = 22100 nM T34099 CIGT04 11974958 Ki = 15900 nM T34099 C75QYG 11974959 Ki = 15800 nM T34099 C2YSR1 11974960 Ki = 11600 nM T34099 C29SWL 11974962 Ki = 20500 nM T34099 CFWI46 11975081 Ki = 2800 nM T34099 CMA18W 24971348 IC50 = 12200 nM T34099 C9BNM3 44405920 Ki = 43 nM T34099 CAM0K8 44405936 Ki > 500000 nM T34099 CO80QU 44405937 Ki = 850 nM T34099 C7FDU0 44405957 Ki = 178000 nM T34099 CRH2Q5 44406028 Ki = 127500 nM T34099 C90MUA 44406029 Ki > 500000 nM T34099 CT4MB6 44406046 Ki > 500000 nM T34099 CHY94P 44406068 Ki > 500000 nM T34099 CB2ZN7 44406070 Ki > 500000 nM T34099 CM9BY6 44406112 Ki = 12000 nM T34099 CCFZ59 44406113 Ki = 6000 nM T34099 CP1LT7 44406115 Ki = 109000 nM T34099 CT6X5P 44453186 Ki = 42800 nM T34099 C58XAZ 44453217 Ki = 82900 nM T34099 CHG0B3 73346535 Ki = 15600 nM T34099 C2A7LY 73354076 Ki = 4900 nM T34099 CRZ62F 73355036 Ki = 750 nM T34099 C1LTY5 73669796 IC50 = 22600 nM T34099 COW4Q7 118714511 IC50 = 3300 nM T34099 C47CKX 118717692 Ki = 4200 nM T34099 C9U0PE 127039493 IC50 = 3800 nM T34099 C1ICT0 127042988 IC50 = 400 nM T34099 CLPO54 154730831 IC50 = 5950 nM T34099 CJZP48 155511221 IC50 = 2300 nM T34099 C5UIX3 155511566 Ki = 300 nM T34099 C1NB5L 155514143 Ki = 300 nM T34099 CM3EJ2 155514596 IC50 = 990 nM T34099 C9M6NW 155515181 IC50 = 4700 nM T34099 C9P1OZ 155519612 IC50 = 1500 nM T34099 CMPN52 155521341 IC50 = 66000 nM T34099 C4QG6L 155522643 IC50 = 16400 nM T34099 C5YV2O 155523279 IC50 = 1700 nM T34099 CK8BS9 155524027 IC50 >= 20000 nM T34099 C7B6QK 155529022 IC50 = 2800 nM T34099 C1R9WH 155530803 IC50 = 1300 nM T34099 C30KYG 155534021 IC50 = 600 nM T34099 CBFP13 155534394 Ki = 300 nM T34099 CLWZ89 155536763 IC50 = 3000 nM T34099 C3URK8 155540339 IC50 > 10000 nM T34099 C8LYT1 155541369 IC50 = 25000 nM T34099 CLH1M8 155541572 Ki = 300 nM T34099 CH36QX 155541714 IC50 = 4100 nM T34099 C4OA7N 155541751 IC50 = 9500 nM T34099 CH4ME8 155542788 IC50 = 9100 nM T34099 CZRJ39 155545268 IC50 = 17700 nM T34099 CW4Y2J 155547311 IC50 = 31800 nM T34099 CUTP53 155548725 IC50 = 1900 nM T34099 C07SZF 155549047 IC50 > 20000 nM T34099 CR9I3F 155551697 IC50 = 6300 nM T34099 CF7EN4 155552740 IC50 = 15900 nM T34099 C2WJI0 155553086 IC50 = 1600 nM T34099 CPA7M1 155553985 IC50 = 2500 nM T34099 CH46TY 155555205 IC50 = 48200 nM T34099 C3DZ2G 155556902 IC50 > 20000 nM T34099 CR6L5Y 155559044 IC50 = 12400 nM T34099 CBG94S 155559399 IC50 = 3600 nM T34099 C0X6BV 155560697 IC50 = 2700 nM T34099 C2RBV0 155562048 IC50 = 121900 nM T34099 CY67CA 155567733 IC50 > 20000 nM T51407 CV24FH 10228 IC50 = 1600 nM T51407 CP4BA8 4496130 IC50 > 25000 nM T51407 C4OG7Z 6917907 IC50 = 1 nM T51407 C4N7XP 45258492 IC50 = 10 nM T51407 CB1RT5 46871912 IC50 = 6400 nM T51407 CVB1Z2 134216299 IC50 = 1500 nM T51407 C75PJO 137650531 IC50 = 25 nM T51407 C6M9EW 155514111 IC50 = 151 nM T51407 D03ZMQ 323 IC50 > 25000 nM T51407 D0U4BB 10748 IC50 > 25000 nM T28213 D0F1LZ 176 IC50 = 120000 nM T28213 D0TA4A 57520598 IC50 = 9 nM T28213 CXR20P 16197 IC50 > 100000 nM T28213 CZN6S9 743974 EC50 > 31622.78 nM T28213 CAVX48 847243 IC50 = 100000 nM T28213 CJ84KX 854190 IC50 > 100000 nM T28213 CK42CY 2397905 IC50 = 800 nM T28213 CUTA28 2520490 IC50 = 2100 nM T28213 C9XR3B 4964042 IC50 = 5200 nM T28213 CX6TJ9 8713297 IC50 > 100000 nM T28213 C9AC6X 9095896 IC50 = 1400 nM T28213 CJ7P8K 12898176 IC50 > 100000 nM T28213 C6VY0J 25479840 IC50 = 56000 nM T28213 C3RCS1 29369661 IC50 = 12000 nM T28213 CDHR65 36477073 IC50 = 1900 nM T28213 CIH5B8 39725404 IC50 = 2000 nM T28213 CBM9S0 46225340 IC50 = 84000 nM T28213 CZB95H 46225341 IC50 > 100000 nM T28213 CV4R1N 46226103 IC50 > 100000 nM T28213 CK8R1G 46226104 IC50 > 100000 nM T28213 CF4KB5 46226105 IC50 > 100000 nM T28213 C9B7SW 46226106 IC50 = 11000 nM T28213 CS6TG2 46226107 IC50 > 100000 nM T28213 CAN53J 46226141 IC50 > 100000 nM T28213 CU8ZM9 46226142 IC50 = 49000 nM T28213 CO9IT1 46226143 IC50 = 1400 nM T28213 CU5H2Y 46226144 IC50 = 1100 nM T28213 CDN5O3 46226145 IC50 = 1300 nM T28213 C8NES0 46226146 IC50 = 53000 nM T28213 CB0W4G 46226160 IC50 = 5700 nM T28213 C4V1LI 46226161 IC50 = 2300 nM T28213 CBH37G 46226162 IC50 = 25000 nM T28213 C6AP1K 46226163 IC50 = 2000 nM T28213 CDV16B 46226164 IC50 = 20000 nM T28213 C58PQO 46226177 IC50 = 100000 nM T28213 C8BHC4 46226178 IC50 = 100000 nM T28213 C9NUX4 46226179 IC50 = 36000 nM T28213 CUD0N1 46226180 IC50 = 57000 nM T28213 CAWB03 46226182 IC50 = 3000 nM T28213 CKA1M0 46226234 IC50 = 4300 nM T28213 C8XMZ6 46226235 IC50 = 17000 nM T28213 C1HKP5 46226236 IC50 = 7900 nM T28213 C7VCJ1 46226237 IC50 > 100000 nM T28213 CBA4T5 46226251 IC50 = 1800 nM T28213 CC4ZU3 46226253 IC50 = 700 nM T28213 C7KPT1 46226254 IC50 = 1500 nM T28213 CA6GS0 46226255 IC50 = 2000 nM T28213 CBN9S3 46226271 IC50 = 79000 nM T28213 CIGN56 46226272 IC50 = 71000 nM T28213 CVYN91 46226273 IC50 = 700 nM T28213 C09JLE 46226274 IC50 = 1000 nM T28213 C52URH 46226275 IC50 = 700 nM T28213 C3WKV7 46226290 IC50 = 1500 nM T28213 CJ7R9Z 46226291 IC50 = 1500 nM T28213 CG1A6V 46226292 IC50 = 500 nM T28213 CFT1U4 46226293 IC50 = 3400 nM T28213 C4L5JT 46226294 IC50 = 700 nM T28213 C1H3VO 46226295 IC50 = 25000 nM T28213 CPST67 46226308 IC50 = 1600 nM T28213 CI64VJ 46226309 IC50 = 1600 nM T28213 C3LG4H 46226310 IC50 = 3800 nM T28213 C4KS9Q 46226311 IC50 = 2400 nM T28213 C7BUZ6 46226312 IC50 = 1200 nM T28213 CQ5AJ3 46226333 IC50 = 46000 nM T28213 C49TEB 46226334 IC50 = 5000 nM T28213 CUI9Z1 46226335 IC50 = 5500 nM T28213 CLM46T 46226336 IC50 = 1200 nM T28213 CC78FP 46226337 IC50 = 600 nM T28213 CZ7T2P 46226338 IC50 = 8800 nM T28213 CA2I8B 46226355 IC50 = 170000 nM T28213 C1RZ3C 46226356 IC50 = 1100 nM T28213 C4DF5S 46226357 IC50 > 100000 nM T28213 CLYW04 46226358 IC50 = 50000 nM T28213 CD6NH8 46226359 IC50 > 100000 nM T28213 CKCR29 46226360 IC50 = 1500 nM T28213 CX6V4F 46226361 IC50 = 5000 nM T28213 CFBQ37 46226382 IC50 = 8500 nM T28213 C7I1UX 46226383 IC50 = 1100 nM T28213 C52QKP 46226384 IC50 > 100000 nM T28213 CY72SF 46226385 IC50 = 16000 nM T28213 C7EK2Y 46226386 IC50 = 45000 nM T28213 CVG2N4 46226436 IC50 > 100000 nM T28213 CL4JK3 46235794 EC50 = 100 nM T28213 CZ7U2W 46869922 EC50 > 10000 nM T28213 C50TDB 53302677 EC50 = 12.59 nM T28213 C6NIF3 67072752 EC50 > 10000 nM T28213 CCBI82 67209218 EC50 = 31.62 nM T28213 CA6O4J 67209297 EC50 = 199.53 nM T28213 CKE6F1 67209751 EC50 = 25.12 nM T28213 COHA70 67210172 EC50 = 31.62 nM T28213 C5Y0HW 67258265 Ki = 478.63 nM T28213 C5R0UC 68175329 IC50 = 7614 nM T28213 CS6KN0 68175794 IC50 = 10000 nM T28213 CS8BA7 68175817 IC50 = 429 nM T28213 C95WQZ 68175946 IC50 = 7820 nM T28213 CB78RL 68175950 IC50 > 10000 nM T28213 CK26DU 68175951 IC50 = 142 nM T28213 CSX58Z 68176013 IC50 = 473 nM T28213 CKSV36 68176091 IC50 = 1208 nM T28213 CAMH36 68176095 IC50 = 442 nM T28213 CZ3AC1 68176096 IC50 = 1584 nM T28213 CAT68L 68176100 IC50 = 510 nM T28213 CWL40T 68176101 IC50 = 3350 nM T28213 CXOG84 68176356 IC50 = 158 nM T28213 C0AZQ7 68176357 IC50 = 245 nM T28213 CX2K5O 70556487 IC50 = 1498 nM T28213 CGB49J 70556496 IC50 = 179 nM T28213 CUZ9N7 70556713 IC50 = 36 nM T28213 CZ7L0W 70556743 IC50 = 5005 nM T28213 COEH02 70556816 IC50 = 123 nM T28213 CUE02Q 70556905 IC50 = 347 nM T28213 CCS1R7 70556909 IC50 = 95 nM T28213 CPHQ85 70557254 IC50 = 321 nM T28213 CR87AK 70557652 IC50 > 10000 nM T28213 C9DOH0 70557757 IC50 = 3350 nM T28213 CJ5K8L 70557795 IC50 = 63 nM T28213 C02ZFH 70557810 IC50 = 500 nM T28213 C5P6DV 70557843 IC50 = 42 nM T28213 CRJ8I5 70557930 IC50 = 57 nM T28213 C4HOZ7 70558275 IC50 = 115 nM T28213 CQHJ02 70558376 IC50 = 278 nM T28213 C8KDN7 70558482 IC50 = 5045 nM T28213 CCNM46 70558485 IC50 = 317 nM T28213 CH37FQ 70558983 IC50 = 781 nM T28213 CG7O4S 70559021 IC50 = 551 nM T28213 C2M0PX 70559086 IC50 = 36 nM T28213 CRIA87 70559096 IC50 = 361 nM T28213 C7G1JL 70559113 IC50 = 118 nM T28213 CSBO56 70559551 IC50 = 256 nM T28213 CVZ41J 70559574 IC50 = 663 nM T28213 C5GSE9 70559585 IC50 = 579 nM T28213 CU3S2C 70559604 IC50 = 25 nM T28213 C5R3UA 70559626 IC50 = 711 nM T28213 CXP0N5 70561343 IC50 = 130 nM T28213 CMWJ75 70562873 IC50 = 85 nM T28213 CV0U9B 70564643 IC50 = 63 nM T28213 CS18MW 70564780 IC50 = 48 nM T28213 CMQ26I 70565254 IC50 = 156 nM T28213 CW0S3G 70566934 IC50 = 90 nM T28213 CE2YV9 77904272 IC50 = 1144 nM T28213 CA24JF 86803193 EC50 > 10000 nM T28213 CNQ59Y 86803224 EC50 > 10000 nM T28213 C7NW3E 88757504 IC50 = 2853 nM T28213 CU3E2R 89894240 IC50 = 116 nM T28213 CG1MH5 89894269 IC50 = 227 nM T28213 C8H6MU 89894353 IC50 = 261 nM T28213 CM72RF 89894379 IC50 = 166 nM T28213 CQ18OE 89900321 IC50 = 1434 nM T28213 CR4X9D 89900324 IC50 > 10000 nM T28213 COWA02 89900327 IC50 = 274 nM T28213 C79QFE 89900346 IC50 = 4673 nM T28213 C60ATU 89900347 IC50 = 247 nM T28213 C4M0NO 89900348 IC50 = 4469 nM T28213 CT0A4L 89900352 IC50 = 143 nM T28213 CO3L0F 89900356 IC50 = 5002 nM T28213 C6GA0I 89900361 IC50 = 388 nM T28213 C27CER 89900365 IC50 = 76 nM T28213 C6LS4P 89900371 IC50 = 263 nM T28213 CNQ2I6 89900378 IC50 = 76 nM T28213 CPH7M6 89901463 IC50 = 44 nM T28213 C13XHQ 117898634 EC50 = 25.12 nM T28213 COS8V6 117898644 EC50 = 25.12 nM T28213 CH1KX8 117898651 EC50 = 25.12 nM T28213 C72IDW 118719384 IC50 = 10000 nM T28213 CRD35S 118719385 IC50 = 10000 nM T28213 CQY80O 118719609 IC50 = 337 nM T28213 C1F9SH 118719610 IC50 = 5800 nM T28213 C1E9ZS 118719611 IC50 = 3350 nM T28213 C4Y7MD 118719612 IC50 = 3350 nM T28213 CZY79J 118719613 IC50 > 10000 nM T28213 C9DR3H 118719614 IC50 > 10000 nM T28213 CJ2A6H 118719615 IC50 > 10000 nM T28213 CJ15RO 118719616 IC50 > 10000 nM T28213 CK24VI 118719617 IC50 = 3350 nM T28213 C17XBZ 118719618 IC50 > 20000 nM T28213 C1Y8QK 118719621 IC50 > 10000 nM T28213 CBVD50 118719622 IC50 > 10000 nM T28213 CK0IY7 118719623 IC50 > 10000 nM T28213 C89JDQ 118719624 IC50 > 10000 nM T28213 CQE20H 118719625 IC50 > 10000 nM T28213 CXKQ09 122184686 EC50 > 10000 nM T28213 C6OPM1 127048827 EC50 > 10000 nM T28213 CH9S7P 127048842 EC50 > 10000 nM T28213 C6V3FP 127050770 EC50 > 10000 nM T28213 CE94RI 127051658 EC50 > 10000 nM T28213 CPBG95 134136959 EC50 > 10000 nM T28213 CJ30RW 134141489 EC50 > 10000 nM T28213 CY3ZF0 134146590 EC50 > 10000 nM T28213 CAG0Y1 134151150 EC50 > 10000 nM T28213 C7MF0A 137633536 EC50 = 25312 nM T28213 CBG58K 137659266 EC50 > 10000 nM T28213 CVP72S 138319694 EC50 = 77.62 nM T28213 CVHA04 145949561 EC50 = 2187.76 nM T28213 CAS97Y 145949591 EC50 = 4786.3 nM T28213 C9W8JQ 145949794 EC50 = 316.23 nM T28213 CGD75I 145950070 EC50 = 1659.59 nM T28213 CD8U0N 145951076 EC50 = 1445.44 nM T28213 CV94XU 145951370 EC50 = 3981.07 nM T28213 C0YOS2 145951537 EC50 = 12.59 nM T28213 CY58OM 145951986 Ki = 338.84 nM T28213 CA7DQ5 145952068 EC50 = 2238.72 nM T28213 C2E9UZ 145952174 EC50 = 2089.3 nM T28213 CR45WT 145952606 EC50 = 3981.07 nM T28213 CJ6C1Q 145953603 EC50 = 1023.29 nM T28213 CQPL24 145953626 Ki = 977.24 nM T28213 CC80KI 145953670 EC50 = 151.36 nM T28213 C9CH2Y 145954073 EC50 = 2818.38 nM T28213 C0J9ZB 145954381 EC50 = 20892.96 nM T28213 CY5PD8 145954653 EC50 = 1348.96 nM T28213 CM8W6H 145955080 EC50 = 812.83 nM T28213 CI43WX 145956912 EC50 = 4466.84 nM T28213 CY95MW 145957026 EC50 = 7079.46 nM T28213 CA7ZP3 145957346 EC50 = 933.25 nM T28213 C4VQ6G 145958427 EC50 = 35481.34 nM T28213 C3URD2 145958672 EC50 = 912.01 nM T28213 CT5JH3 145959365 EC50 = 2238.72 nM T28213 CE53LG 145959580 EC50 = 4786.3 nM T28213 C5TME3 145962491 EC50 = 213.8 nM T28213 CKI2M4 145971768 EC50 = 1288.25 nM T28213 D05UBB 46226252 IC50 = 500 nM T28213 D07ITP 854189 EC50 = 100 nM T28213 D08ZYC 11595431 EC50 < 50118.72 nM T28213 D0I3EQ 4307629 IC50 = 800 nM T28213 D0S5BG 1032 EC50 = 250000 nM T14894 CDT9G3 11467504 IC50 = 29.5 nM T14894 CDY2W5 49796910 IC50 = 17.7 nM T14894 CGY3W2 71471109 IC50 = 590 nM T14894 CANH70 71716242 IC50 = 420 nM T14894 C40WIR 71718085 IC50 = 3300 nM T14894 CU75VK 71719897 IC50 = 130 nM T14894 CBV6F1 71720507 IC50 = 2670 nM T14894 D0Y5IQ 44255320 IC50 = 5000 nM T79307 D0E3TC 44259 IC50 = 8.95 nM T79307 C5AGH6 6604378 EC50 = 263.1 nM T79307 C60XTH 59225335 IC50 = 2.9 nM T79307 CX3U6H 63043775 IC50 = 22400 nM T79307 CV63UL 67240318 IC50 > 10000 nM T79307 COG97V 86346643 IC50 = 5.3 nM T79307 C19SVO 91827516 IC50 = 120 nM T79307 CD7U6E 92044402 IC50 = 108 nM T79307 CL57JX 122186227 IC50 = 67 nM T79307 CH91ON 129245363 IC50 > 10000 nM T79307 CEYK58 129245795 IC50 = 28 nM T79307 CQJK71 129246093 IC50 = 980 nM T79307 CCF8W2 129261617 IC50 = 1640 nM T79307 C2LWZ1 129318964 IC50 > 10000 nM T79307 C34XMQ 131801113 EC50 = 18.94 nM T79307 C6OP3W 135397688 IC50 = 3050 nM T79307 CM07EU 145714274 IC50 = 9 nM T79307 C9ISH6 145925685 IC50 = 7930 nM T79307 CX9M5Y 145949246 IC50 = 330 nM T79307 CK3Q4O 145950368 IC50 = 560 nM T79307 CGD13Y 145950439 IC50 = 4230 nM T79307 C43FMJ 145950943 IC50 = 4940 nM T79307 C8PJ9Q 145951585 IC50 = 840 nM T79307 CA0C5V 145952095 IC50 = 2220 nM T79307 C4O2YR 145952213 IC50 = 2730 nM T79307 CKC01D 145952842 IC50 > 33000 nM T79307 CWK06E 145952967 IC50 = 110 nM T79307 C0HI8L 145953121 IC50 = 18100 nM T79307 C2D0JL 145953281 IC50 = 1490 nM T79307 CY6C7Z 145953376 IC50 = 11 nM T79307 CZXS75 145954619 IC50 = 183 nM T79307 CRLB02 145954690 IC50 = 589 nM T79307 CBM21S 145955762 IC50 = 670 nM T79307 CEAY65 145955845 IC50 = 45 nM T79307 CSEO43 145957285 IC50 = 1830 nM T79307 CYQ41D 145957913 IC50 = 239 nM T79307 CC2XD6 145959005 IC50 = 315 nM T79307 CHQK46 145959382 IC50 = 24 nM T79307 CJI0R3 145959412 IC50 = 477 nM T79307 CZ06DA 145959556 IC50 = 288 nM T79307 CXY2R7 145959677 IC50 = 242 nM T79307 CBD17G 145962774 IC50 = 45 nM T79307 CIO25W 145966088 EC50 = 54.84 nM T79307 CLB0W7 145966392 EC50 = 40.8 nM T79307 CV4IW9 145971727 IC50 = 840 nM T79307 CKJ0C1 145973347 IC50 = 416 nM T79307 CL9J0U 145973629 IC50 = 368 nM T79307 CP53VU 145974061 IC50 = 40 nM T79307 C4PCO0 145978715 EC50 = 24.14 nM T79307 C7CH9V 146014951 IC50 = 263 nM T79307 C2MD1Q 155513187 IC50 > 10000 nM T79307 CZ0WO7 155523990 IC50 = 416 nM T79307 CHD09S 155543566 IC50 = 368 nM T79307 D06ZIO 44464263 IC50 = 45 nM T79307 D0RG0Z 10077147 IC50 = 87 nM T99912 CC62AF 161166 Ki = 4280 nM T99912 CT9U1P 9794338 Ki = 100 nM T99912 CZ96MS 18368983 Ki = 70 nM T99912 CCX6W8 44322715 Ki = 8800 nM T99912 C60VNB 44322835 Ki = 70 nM T99912 CQ4R2L 44322939 Ki = 880000 nM T99912 CD9NO7 10888792 Ki = 23400 nM T99912 D05JZS 450268 Ki = 60000 nM T65200 D0PQ3G 3440 IC50 = 3760 nM T65200 D02ENG 6918651 IC50 = 3341 nM T65200 D05WCI 11670435 Ki = 9 nM T65200 D08VSQ 59336911 IC50 = 3 nM T65200 D0B5HF 44476893 IC50 = 1.7 nM T65200 D0O1ZI 25006684 IC50 = 2 nM T65200 D0R8IU 24946280 IC50 = 7 nM T65200 D0S2PD 42634627 Ki = 0.9 nM T65200 D0T8QB 14982 EC50 = 10 nM T65200 D07EBU 135565424 IC50 = 0.000975 ug.mL-1 T65200 D07FHW 23725123 Ki < 1 nM T65200 CHN16X 81439 IC50 > 100000 nM T65200 CDM6C4 92730 IC50 = 630 nM T65200 C7JEN0 94320 IC50 = 800 nM T65200 C2O8KM 101788 IC50 = 1160 nM T65200 CFG6D1 111253 IC50 = 619 nM T65200 CPY37Z 229604 IC50 > 100000 nM T65200 CRU5Q4 257864 IC50 = 20000 nM T65200 C8W3LH 286220 IC50 > 100000 nM T65200 C7TYH9 585624 IC50 = 676 nM T65200 CH2D1M 655951 IC50 = 23600 nM T65200 CB68LK 656335 IC50 > 100000 nM T65200 CKZ53V 658196 IC50 = 2816 nM T65200 C0WM4A 686457 IC50 = 877 nM T65200 CX2W4R 722461 IC50 = 628 nM T65200 C9REL7 723651 IC50 = 266 nM T65200 CY2SM6 735815 IC50 > 1000 nM T65200 CD8G9Y 755284 Ki = 84 nM T65200 CSU6P2 777284 IC50 > 100000 nM T65200 CIV19J 798754 IC50 = 53000 nM T65200 C2AK7U 812578 IC50 = 435 nM T65200 CR6F9A 812579 IC50 = 326 nM T65200 CMT1K9 870990 IC50 = 860 nM T65200 C1R8KM 891290 IC50 = 86 nM T65200 COF9Z7 984480 IC50 = 647 nM T65200 C2DEU1 984483 IC50 = 1672 nM T65200 C27WFR 984493 IC50 = 15900 nM T65200 C04XRN 984541 IC50 = 1208 nM T65200 C2Q8YS 1000718 IC50 = 3740 nM T65200 CFUM35 1035303 IC50 = 4580 nM T65200 C4TJ7S 1041738 IC50 = 42 nM T65200 CU28EL 1041872 IC50 = 3570 nM T65200 CUFT92 1153922 IC50 = 160 nM T65200 C9X8TL 1203924 IC50 = 4000 nM T65200 C15LUS 1217734 IC50 = 6280 nM T65200 C9OI2P 1268251 IC50 = 507 nM T65200 CKV04E 1277351 IC50 = 106 nM T65200 C47WPI 1289623 IC50 = 1031 nM T65200 C4KCW8 1418612 IC50 = 30 nM T65200 C5QC7L 1437062 IC50 = 3610 nM T65200 CX9H0V 1437818 IC50 = 3410 nM T65200 CMWC23 1437824 IC50 = 4200 nM T65200 CER5N9 1437832 IC50 = 7440 nM T65200 CJP27D 1437837 IC50 = 21800 nM T65200 CUE8F2 1437841 IC50 = 6020 nM T65200 CJK9B1 1438038 IC50 = 15800 nM T65200 CO4C7Q 1438157 IC50 = 6890 nM T65200 CC6U5G 1438163 IC50 = 21900 nM T65200 CPY8W1 1438312 IC50 = 7500 nM T65200 CFZ8C1 1462195 IC50 = 6400 nM T65200 CF23IT 1462198 IC50 = 4200 nM T65200 CG93IP 1475852 IC50 = 12 nM T65200 C7D6PV 1475853 IC50 = 4 nM T65200 C8UQT9 1484979 IC50 = 16 nM T65200 CN2X0Q 1484980 IC50 = 456 nM T65200 C4UJO6 1484981 IC50 = 14 nM T65200 CFB1L9 1551384 IC50 = 263 nM T65200 CW72DZ 1551387 IC50 = 17393 nM T65200 CR8M3N 1562409 IC50 = 690 nM T65200 CD93XP 1717478 IC50 = 770 nM T65200 C5NDC2 1732003 IC50 = 2100 nM T65200 CC40IA 1909086 IC50 = 195 nM T65200 CJR97X 2200386 IC50 = 1215 nM T65200 CV7P3Z 2206056 IC50 = 95 nM T65200 COF86A 2214845 IC50 = 1733 nM T65200 CF4CU8 2738343 IC50 = 28.8 nM T65200 CA09DR 2741409 IC50 > 1000 nM T65200 COF0Q8 2741412 IC50 = 61 nM T65200 C8NG7R 2741589 IC50 = 262 nM T65200 C50CFU 2741649 IC50 = 32.7 nM T65200 C2ZUN0 2747154 IC50 = 45 nM T65200 CRZ30P 2795955 IC50 = 3.7 nM T65200 CQYV95 2804743 IC50 = 41.3 nM T65200 CC6J2D 2805256 IC50 = 403 nM T65200 C4ZIH1 2807133 IC50 = 102.4 nM T65200 CW67OP 2827468 IC50 = 700 nM T65200 C9JT7I 2851184 IC50 = 1860 nM T65200 C38VJU 2882437 IC50 = 80 nM T65200 CCA57W 2901354 IC50 = 14600 nM T65200 CQD6O3 2903292 IC50 = 5600 nM T65200 CQ2GS3 2950639 IC50 = 2030 nM T65200 C34FUY 2953793 Ki = 175 nM T65200 C8JWK2 2998753 IC50 = 7200 nM T65200 C89MEO 2999452 IC50 > 100000 nM T65200 CT9WZ1 3036892 IC50 > 1000 nM T65200 C2E5ND 3143222 IC50 = 260 nM T65200 C3B7LM 3146235 IC50 = 58.1 nM T65200 C9POC1 3502039 IC50 > 100000 nM T65200 C85DYG 3604343 IC50 = 20 nM T65200 C1F4ZY 3812801 Ki = 108 nM T65200 C3LSG7 3860166 IC50 = 234 nM T65200 C1PS0T 4119853 IC50 > 100000 nM T65200 CM3RB8 4332595 IC50 = 35500 nM T65200 C1UGY7 4385295 IC50 = 61 nM T65200 CHP86W 4432326 IC50 = 48000 nM T65200 CJ4HF1 4454335 IC50 = 5870 nM T65200 CWP9Y7 4570352 IC50 > 100000 nM T65200 CV0H2K 4592745 IC50 = 90000 nM T65200 CI9KQ2 4982676 Ki = 48 nM T65200 C86WNE 5060832 IC50 = 44000 nM T65200 C0L1UN 5151632 IC50 > 100000 nM T65200 CHR5O7 5296322 IC50 = 679 nM T65200 CEC9O8 5349980 IC50 = 14800 nM T65200 C1OZS6 5436342 IC50 = 31 nM T65200 CX2O4S 5715869 IC50 = 66.7 nM T65200 CZM01L 5946474 IC50 = 388 nM T65200 CWF94G 6048619 IC50 = 97 nM T65200 CK1W2Z 6227694 IC50 = 254 nM T65200 CDFX51 6872813 IC50 = 1850 nM T65200 C9PO8Y 6874186 IC50 > 50000 nM T65200 CPT5Y6 6918663 IC50 = 28.4 nM T65200 C3O1TA 6918868 IC50 = 3200 nM T65200 CJQ1K0 7312225 IC50 = 980 nM T65200 CNW9Q0 7509285 IC50 = 19 nM T65200 C7KQA1 8178360 IC50 = 520 nM T65200 C8J5PX 9107173 IC50 = 37 nM T65200 CKU73M 9114624 IC50 = 47000 nM T65200 C84RBQ 9797661 IC50 = 5 nM T65200 CY2K5B 9823394 IC50 = 1.2 nM T65200 CHV1E3 9975108 IC50 = 2 nM T65200 CSL50G 9975639 IC50 = 2.7 nM T65200 CDZ92L 9998483 IC50 = 0.28 nM T65200 CBUP07 10018475 IC50 = 1 nM T65200 C0I6WB 10040175 IC50 = 1 nM T65200 CU1W4M 10040176 IC50 = 2 nM T65200 C4L0HV 10043410 IC50 = 5 nM T65200 CXV5Q2 10046202 IC50 = 9060 nM T65200 CA4SJ7 10064183 IC50 = 8 nM T65200 C9IH1Y 10065028 IC50 = 5 nM T65200 C5LKO8 10085885 IC50 = 2 nM T65200 CW6KU4 10250720 IC50 = 1.995 nM T65200 CO0H7A 10250842 IC50 = 2.3 nM T65200 COT1X3 10308303 IC50 = 7.8 nM T65200 C2LWK5 10315044 IC50 = 5 nM T65200 C0QH6L 10335644 IC50 = 43 nM T65200 C7IUQ6 10335880 IC50 = 1 nM T65200 CI64PJ 10340916 IC50 = 11 nM T65200 CL5X6K 10355633 IC50 = 8 nM T65200 CTLN27 10357519 IC50 = 2 nM T65200 CTU13Q 10357992 IC50 = 2 nM T65200 CWKP54 10359991 IC50 = 2 nM T65200 CEO4C7 10360107 IC50 = 32 nM T65200 CUL28X 10380007 IC50 = 1 nM T65200 CF4NL2 10381554 IC50 = 15 nM T65200 CR4V3G 10402262 IC50 = 2 nM T65200 C65EQT 10403095 IC50 = 13 nM T65200 CV8K3E 10446474 IC50 = 1 nM T65200 CQ9X4Y 10446475 IC50 = 1 nM T65200 CYI70T 10447474 IC50 = 2 nM T65200 CS06QG 10452320 Ki = 14 nM T65200 CA89WN 10470037 IC50 = 3 nM T65200 C8HPS1 10471798 IC50 = 2 nM T65200 C6LJI0 10473292 IC50 = 2.7 nM T65200 CXH39G 10474399 IC50 = 3 nM T65200 CJR1T6 11033292 IC50 = 240 nM T65200 C3X0AC 11155482 IC50 = 3 nM T65200 C0C6KD 11190936 IC50 = 1157 nM T65200 CN97TW 11191097 IC50 = 0.9 nM T65200 CX64TS 11199934 IC50 < 1 nM T65200 CP9Z1V 11225445 IC50 = 0.4 nM T65200 CD3H7R 11232699 IC50 = 190 nM T65200 C1PKI0 11257147 IC50 = 8912.51 nM T65200 CW1T5X 11259177 IC50 = 13 nM T65200 CH12WK 11278558 IC50 = 110 nM T65200 CP9O5R 11280328 IC50 = 2300 nM T65200 C28ZPF 11280485 IC50 = 170 nM T65200 CH85OD 11319723 IC50 = 2810 nM T65200 CN94OC 11329380 IC50 = 1.1 nM T65200 CD7V8S 11353668 IC50 = 52 ug.mL-1 T65200 C1IU3K 11375115 IC50 = 0.5 nM T65200 C8FQ9B 11375180 IC50 = 144 nM T65200 CI0K2V 11420598 IC50 = 0.5 nM T65200 C1YV6P 11442292 IC50 = 1.7 nM T65200 CH6X2L 11478011 IC50 = 1.2 nM T65200 CS0P1Q 11478969 IC50 = 3840 nM T65200 CR4I9H 11484764 IC50 = 35 nM T65200 CM02LZ 11494480 IC50 = 1.3 nM T65200 CE2ZN7 11495528 IC50 = 5.012 nM T65200 CN08AP 11495851 Ki = 8 nM T65200 CC8ZQ5 11502331 IC50 = 1071.52 nM T65200 CLT1Z9 11502804 Ki = 4 nM T65200 C76STL 11504178 Ki = 13 nM T65200 C19BYP 11505338 IC50 = 310 nM T65200 CHW7L1 11510573 Ki = 6 nM T65200 C24TMY 11515715 IC50 = 4.4 nM T65200 CD7AE3 11522916 IC50 = 3.1 nM T65200 CT3A4Z 11523500 IC50 = 4.6 nM T65200 CE40MU 11524868 IC50 = 54 nM T65200 C8NP4Y 11526147 IC50 = 1.995 nM T65200 C6E5LW 11532049 IC50 = 40.74 nM T65200 C4KU0S 11532178 IC50 = 6.026 nM T65200 CPW4T6 11532312 IC50 = 43.65 nM T65200 CG1HB5 11533520 Ki = 18 nM T65200 C1UYS4 11538562 IC50 = 0.8 nM T65200 C57DMG 11538907 IC50 = 104.71 nM T65200 CXYJ80 11538963 IC50 = 2.3 nM T65200 CZE42S 11540388 IC50 = 27 nM T65200 CN1A6F 11540493 Ki = 6 nM T65200 CKY2F7 11544921 IC50 = 2.6 nM T65200 C3LVE2 11545617 IC50 = 21.88 nM T65200 C16HDK 11545694 Ki = 287 nM T65200 CD17CO 11551576 IC50 = 832 nM T65200 CP8L9K 11552169 IC50 = 5.012 nM T65200 CCT0Q7 11552781 IC50 = 6 nM T65200 CA25ZF 11555218 Ki = 7 nM T65200 CC73PF 11565519 IC50 = 1.2 nM T65200 CEM8Q3 11565865 IC50 = 30 nM T65200 C8WG6Z 11574633 IC50 = 2.7 nM T65200 CJ58XB 11576524 Ki = 7 nM T65200 C53IBR 11581555 IC50 = 5.2 nM T65200 C8YO0H 11587817 IC50 = 5.8 nM T65200 CLW6G9 11589149 IC50 = 2.9 nM T65200 CTJ1I6 11589339 IC50 = 1096.48 nM T65200 C83TBC 11589528 IC50 = 44.67 nM T65200 CZ3MB0 11603067 IC50 = 50.12 nM T65200 CC43XK 11604154 IC50 = 89.13 nM T65200 CKF3J6 11604308 Ki = 5 nM T65200 CS2ZV8 11609013 Ki = 3.6 nM T65200 C81PFA 11609989 IC50 = 2.1 nM T65200 CGD7X9 11610822 IC50 = 6 nM T65200 C5WCZ7 11610825 IC50 = 7943.28 nM T65200 CPV31O 11610957 IC50 = 1584.89 nM T65200 CDL39R 11613794 IC50 = 300 nM T65200 C7KBZ4 11618761 Ki = 4 nM T65200 CB4HL1 11625219 IC50 = 1.3 nM T65200 CW2XN3 11626362 Ki = 8 nM T65200 CXS05L 11627334 Ki = 7 nM T65200 CMF3U5 11634114 Ki = 8 nM T65200 CTI1G0 11638307 IC50 = 2.2 nM T65200 CDL94B 11649095 Ki = 6 nM T65200 CX17LY 11654021 IC50 = 7.943 nM T65200 C3B4SN 11655097 Ki = 26 nM T65200 C1DJ7W 11655188 Ki = 7 nM T65200 CI3SO6 11659479 IC50 = 2.9 nM T65200 C1T6KE 11666874 Ki = 2 nM T65200 C16IKG 11667087 IC50 = 0.03 nM T65200 CCNY17 11669908 IC50 = 294 nM T65200 CFH6G5 11670914 IC50 = 15 nM T65200 CU5TI1 11676805 Ki = 5 nM T65200 CE17ZX 11681796 IC50 = 2 nM T65200 CK6P7Y 11682215 IC50 = 0.98 nM T65200 CVXC54 11682929 IC50 = 18 nM T65200 CK1R3T 11683156 IC50 < 1 nM T65200 C69RWN 11688174 IC50 = 102 nM T65200 CDEP02 11689246 IC50 = 4.3 nM T65200 C1XI5U 11695884 IC50 = 0.32 nM T65200 CJ13XD 11698697 IC50 = 25 nM T65200 C26ITU 11699075 Ki = 17 nM T65200 C2P6SV 11702545 IC50 = 0.98 nM T65200 CTU0H9 11703148 IC50 = 0.98 nM T65200 CK8BF3 11705872 Ki = 8 nM T65200 C4WC9D 11710272 IC50 = 14.13 nM T65200 C4D6YM 11712182 Ki = 14 nM T65200 CR1X5T 11717880 IC50 = 1 nM T65200 C5AT6X 11722880 IC50 = 10 nM T65200 CO32UM 11724534 IC50 = 2 nM T65200 C6TPR1 11739354 IC50 = 289 nM T65200 C4B5XT 11741200 IC50 = 2 nM T65200 CB9WI2 11742158 IC50 = 13 nM T65200 C37IRX 11771845 IC50 = 4 nM T65200 CND4T6 11774173 Ki = 169 nM T65200 CCHL73 11835767 IC50 = 850 nM T65200 C5N4CJ 11835998 IC50 > 10000 nM T65200 CF38GR 11841377 IC50 = 5300 nM T65200 C2XW0P 11853305 IC50 = 172 nM T65200 CZ31IA 12000645 IC50 = 21.4 nM T65200 CIN35F 12002965 EC50 = 327 nM T65200 CHP0A4 12002967 EC50 = 58 nM T65200 CC57SI 12002968 Ki = 4.8 nM T65200 CD4UA7 12003049 EC50 = 184 nM T65200 CIO30R 12003050 EC50 = 1161 nM T65200 CZGJ92 12003051 EC50 = 51 nM T65200 CY9W5R 12003052 EC50 = 936 nM T65200 CS6JO0 12033869 IC50 = 144 nM T65200 CV4HP7 13603965 IC50 = 9120 nM T65200 CY57NQ 13948729 IC50 = 529 nM T65200 C4FKP2 13994830 IC50 = 1236 nM T65200 CQ6UA7 15016062 IC50 = 350 nM T65200 C6EC5N 15204385 IC50 = 130 nM T65200 CJ06RL 15953418 IC50 = 11 nM T65200 CDK52O 15953420 IC50 = 2962 nM T65200 CA8ML0 15953421 IC50 = 34 nM T65200 CM7I6B 15953422 IC50 = 12 nM T65200 C3N7VE 15953424 IC50 = 23 nM T65200 CEYW48 15953464 IC50 = 12 nM T65200 CX80AP 15953467 IC50 = 11 nM T65200 C8F6EP 15953469 IC50 = 143 nM T65200 C3QL4H 15953516 IC50 = 72 nM T65200 C4X1UF 15986762 IC50 = 36 nM T65200 CC0IO7 15987307 IC50 = 9 nM T65200 CY3A6Q 15987396 IC50 = 0.7 nM T65200 C29ACV 15987476 IC50 = 6.6 nM T65200 CA0ZR8 15987477 IC50 = 0.88 nM T65200 CO4BE6 15997991 IC50 = 10 nM T65200 C02YOC 16045371 IC50 = 41 nM T65200 CN2A3D 16045446 IC50 = 116 nM T65200 CUV8G1 16045450 IC50 = 63 nM T65200 C72CQB 16045524 IC50 = 19 nM T65200 C8E6VT 16045526 IC50 = 10 nM T65200 C6QSC4 16045529 IC50 = 9.7 nM T65200 CQY8K7 16045596 IC50 = 9.9 nM T65200 CKW9C7 16045597 IC50 = 9 nM T65200 C19WPN 16045599 IC50 = 13 nM T65200 C7G5PB 16045600 IC50 = 3.1 nM T65200 C5XJY3 16045657 IC50 = 46 nM T65200 CS1XM4 16049788 IC50 = 12.88 nM T65200 COS87Z 16100382 Ki = 5 nM T65200 CTC19G 16100386 Ki = 62 nM T65200 CZ80NG 16100389 Ki = 10 nM T65200 CU9X8E 16100403 Ki = 24 nM T65200 CJO58L 16116998 IC50 = 7 nM T65200 C9HI7G 16118895 IC50 = 10 nM T65200 CT3YW2 16118896 IC50 = 14 nM T65200 CDEZ74 16118897 IC50 = 13 nM T65200 C3IV0E 16118898 IC50 = 7 nM T65200 CF7M3V 16118899 IC50 = 9 nM T65200 C8ZEG9 16118900 IC50 = 4 nM T65200 C2T4IM 16222378 IC50 = 3100 nM T65200 C5UH7K 16299367 IC50 = 1900 nM T65200 CTA73M 16311434 IC50 = 600 nM T65200 CG2ED3 16348684 IC50 = 1500 nM T65200 C1Y0GH 16371048 Ki = 2600 nM T65200 C56EKI 16371051 Ki = 300 nM T65200 CF5E4J 16371339 Ki = 3100 nM T65200 CW5LP8 16377050 Ki = 3500 nM T65200 C13TPH 16721119 Ki = 4 nM T65200 CA9L6H 16724456 IC50 = 37 nM T65200 C2OJC1 16726072 IC50 = 1.6 nM T65200 CHO03N 16742060 IC50 = 120 nM T65200 CAW6P7 16752710 Ki = 190 nM T65200 CK87ZX 16812383 IC50 = 700 nM T65200 CW3E2F 17396226 Ki > 10000 nM T65200 CTDB09 17403222 IC50 = 379 nM T65200 C5JY6A 17407272 IC50 = 1000 nM T65200 C9V1TW 17752924 Ki = 100 nM T65200 CDX4V6 19414526 IC50 = 12.59 nM T65200 C18KDZ 19682724 IC50 = 87 nM T65200 C7M5WN 19684374 IC50 = 32 nM T65200 CGW6I0 20416676 IC50 = 346 nM T65200 CWU4M0 20704168 IC50 > 1000 nM T65200 C69QUM 20724870 IC50 = 27 nM T65200 C51LGI 20724898 IC50 = 9.3 nM T65200 CP7JM8 20724899 IC50 = 1.7 nM T65200 C31VAH 20724901 IC50 = 1 nM T65200 CJU3T5 20724903 IC50 = 2.2 nM T65200 CLX5A8 20724912 IC50 = 1 nM T65200 CQ6CF3 20755069 IC50 = 4.1 nM T65200 C4P3EK 20755074 IC50 = 4 nM T65200 CTRD81 20755103 IC50 < 1 nM T65200 CGNU19 21099751 IC50 = 14.13 nM T65200 CCN9K7 21099775 IC50 = 28.84 nM T65200 COCH32 21099776 IC50 = 46.77 nM T65200 CD1SR0 22591684 IC50 = 3.2 nM T65200 CQ6AO5 22591709 IC50 = 7 nM T65200 CWF51V 22591726 IC50 = 6.1 nM T65200 C9K1DY 23583191 IC50 = 114 nM T65200 CACL45 23634382 IC50 = 108 nM T65200 C9HG7A 23634383 IC50 = 0.5 nM T65200 CB2WV5 23648664 IC50 = 4 nM T65200 CWS12O 23648694 IC50 = 3 nM T65200 CL4VK3 23794291 IC50 = 1470 nM T65200 C5FN6C 24072323 IC50 = 28 nM T65200 CQ46WF 24735746 Ki > 10000 nM T65200 CDS4T7 24744018 IC50 = 5 nM T65200 CEB47A 24744047 IC50 = 16.1 nM T65200 C7HT5Q 24744154 IC50 = 200 nM T65200 CH53FU 24783779 IC50 = 6904 nM T65200 CNFD06 24785815 IC50 = 16 nM T65200 CF7BV4 24785816 IC50 = 85 nM T65200 C9W2KX 24812720 IC50 = 3 nM T65200 CL46CW 24824737 IC50 = 1.5 nM T65200 C3SO6V 24824766 IC50 = 14 nM T65200 CL08VC 24825785 IC50 = 9 nM T65200 CGR84K 24854349 IC50 = 13 nM T65200 C6BV8N 24854350 IC50 > 500000 nM T65200 CEW31B 24856362 Ki = 1.1 nM T65200 CQHV30 24857855 IC50 = 1 nM T65200 C7QU2Z 24883422 IC50 = 1417 nM T65200 C1B5QK 24884555 IC50 = 78 nM T65200 CLYS75 24889741 IC50 = 51 nM T65200 CVD4K7 24889906 IC50 = 5 nM T65200 C6EFK9 24889907 Ki = 50 nM T65200 C5QD7L 24890069 IC50 = 41 nM T65200 C9XUC0 24890070 IC50 = 28 nM T65200 C3A9HI 24890073 IC50 = 51 nM T65200 C6IHL0 24890239 IC50 = 45 nM T65200 C9J2BQ 24895553 IC50 = 1.3 nM T65200 CEV27L 24895554 IC50 = 1.3 nM T65200 C8LYV0 24895658 IC50 = 0.7 nM T65200 CASQ47 24895660 IC50 = 2.6 nM T65200 C2QWU0 24895661 IC50 = 2.4 nM T65200 C1G6DM 24895969 IC50 = 42 nM T65200 C59MRG 24896012 IC50 = 66 nM T65200 C9Z8KO 24896014 IC50 = 66 nM T65200 C8FPH7 24896062 IC50 = 20 nM T65200 CNRO54 24901355 IC50 = 11 nM T65200 CSFG34 24905449 IC50 = 300 nM T65200 CH3YR8 24906056 IC50 = 1300 nM T65200 CFU31W 24906057 IC50 = 500 nM T65200 C49UAN 24906058 IC50 = 9900 nM T65200 C9UE4R 24906059 IC50 = 52 nM T65200 CIW1N9 24906060 IC50 = 68 nM T65200 C72TSQ 24906061 IC50 = 10 nM T65200 CB81TR 24906102 IC50 = 15 nM T65200 CJ4I1H 24906103 IC50 = 13 nM T65200 C26WCT 24906104 IC50 = 21 nM T65200 C9BL7W 24906105 IC50 = 30 nM T65200 CJK4Q1 24906106 IC50 = 490 nM T65200 CY52UI 24906147 IC50 > 10000 nM T65200 CV0PQ2 24906148 IC50 = 61 nM T65200 CQ46LP 24906149 IC50 = 10 nM T65200 CK1ED3 24906190 IC50 = 10 nM T65200 CM6RL4 24906191 IC50 = 28 nM T65200 CYA51J 24906192 IC50 = 11 nM T65200 CQ83BP 24906193 IC50 = 160 nM T65200 CL56ST 24906194 IC50 = 32 nM T65200 C3Z4AJ 24906237 IC50 = 26 nM T65200 C29UYD 24906238 IC50 = 120 nM T65200 C0X8AC 24906239 IC50 = 74 nM T65200 CI2Z0D 24906240 IC50 = 13 nM T65200 CUL9K2 24941247 IC50 = 1.6 nM T65200 C7Y8GV 24944569 IC50 = 2 nM T65200 C4EJ3F 24944723 IC50 = 2.2 nM T65200 C0Q5BI 24944725 IC50 = 13 nM T65200 C4MX5U 24944726 IC50 = 8950 nM T65200 CP35BN 24945154 IC50 = 156 nM T65200 CR8E1G 24945155 IC50 = 24 nM T65200 C97KJC 24945156 IC50 = 7 nM T65200 C29JWS 24945158 IC50 = 16 nM T65200 CQ8H1M 24945160 IC50 = 3 nM T65200 C9ZKU7 24945236 IC50 = 5 nM T65200 C0VLU6 24945237 IC50 = 4 nM T65200 CT8DF6 24945238 IC50 = 12 nM T65200 CIT4D0 24945240 IC50 = 193 nM T65200 CUN93Q 24945241 IC50 = 594 nM T65200 CF5LM1 24945242 IC50 = 63 nM T65200 CSHU94 24945243 IC50 = 204 nM T65200 CO79YV 24945402 IC50 = 160 nM T65200 C57DSQ 24945403 IC50 = 21 nM T65200 C56HDY 24945482 IC50 = 4.9 nM T65200 CP8B6D 24945561 IC50 = 9 nM T65200 C7RI1B 24945563 IC50 = 1 nM T65200 C8ED9K 24945565 IC50 = 0.6 nM T65200 C58VOY 24945566 IC50 = 3 nM T65200 CD6PT4 24945640 IC50 = 20 nM T65200 COV53C 24945641 IC50 = 25 nM T65200 CVIO68 24945642 IC50 = 1 nM T65200 C8HJ0E 24945643 IC50 = 65 nM T65200 CI81ZP 24945724 IC50 = 22 nM T65200 CK5TJ7 24945801 IC50 = 0.8 nM T65200 CHZE54 24946103 IC50 = 96 nM T65200 CKG20D 24946104 IC50 = 140 nM T65200 C90SNX 24946105 IC50 = 220 nM T65200 CX6E2B 24946106 IC50 = 200 nM T65200 CKZ2J4 24946279 IC50 = 160 nM T65200 CZ3GW2 24946456 IC50 = 700 nM T65200 CAY0X5 24946799 IC50 = 2100 nM T65200 CE5K9B 24946802 IC50 = 99 nM T65200 CDXB43 24946979 IC50 = 47 nM T65200 C2PMA0 24946980 IC50 = 120 nM T65200 C2Z6JK 24947160 IC50 = 37 nM T65200 CO4J2S 24947161 IC50 = 38 nM T65200 CFA4I2 24947239 IC50 = 1800 nM T65200 CF07NV 24947347 IC50 = 21 nM T65200 C2BZ0M 24947416 IC50 = 17 nM T65200 CZ02KJ 24947418 IC50 = 9 nM T65200 CC86ZH 24947419 IC50 = 48 nM T65200 C2OYA4 24947420 IC50 = 18 nM T65200 CXLF42 24947421 IC50 = 16 nM T65200 C9DZ1U 24947607 IC50 = 60 nM T65200 CP25EF 24947608 IC50 = 48 nM T65200 CV8UO9 24947610 IC50 = 150 nM T65200 C4NX8M 24947800 IC50 = 160 nM T65200 CE1GR4 24947984 IC50 = 340 nM T65200 C6UYQ4 24948172 IC50 = 8 nM T65200 CBJ67E 24948362 IC50 = 200 nM T65200 CA4RG2 24948552 IC50 = 57 nM T65200 C1RA5T 24948553 IC50 = 8 nM T65200 C54TVH 24948738 IC50 = 12 nM T65200 C3Y9RU 25002426 IC50 = 110 nM T65200 C9ZP3W 25005578 IC50 = 3 nM T65200 C5N2OH 25005580 IC50 = 43 nM T65200 CE1MR4 25005939 IC50 = 21 nM T65200 CYW9J0 25006685 IC50 = 6 nM T65200 C9JZ6W 25006686 IC50 = 9 nM T65200 C5XA3B 25006687 IC50 = 380 nM T65200 C23YDF 25006688 IC50 = 17 nM T65200 C4VNY5 25007063 IC50 = 10 nM T65200 C02KHV 25007064 IC50 = 7600 nM T65200 CM0G6D 25007066 IC50 = 11 nM T65200 C1ILM9 25007438 IC50 = 5 nM T65200 CQUO09 25007441 IC50 = 12 nM T65200 CC3QA7 25007798 IC50 = 4 nM T65200 C0J6SK 25007799 IC50 = 10 nM T65200 CKE0Y4 25007800 IC50 = 190 nM T65200 CU2GL0 25015962 IC50 = 2.2 nM T65200 C3TWB7 25016990 IC50 = 97 nM T65200 CK8L1J 25017526 IC50 = 9 nM T65200 CB8UR4 25017529 IC50 = 1.4 nM T65200 CTI5L0 25017780 IC50 = 62 nM T65200 CT4UF0 25018029 IC50 = 1.4 nM T65200 CQ61PH 25018032 IC50 = 43 nM T65200 C0MVY6 25018527 IC50 = 190 nM T65200 C3G1MS 25019046 IC50 = 64 nM T65200 C82BOU 25019309 IC50 = 0.8 nM T65200 C6HFK4 25019564 IC50 = 34 nM T65200 C56CLP 25063949 IC50 = 68.6 nM T65200 CZNG30 25064398 IC50 = 0.8 nM T65200 CJL38O 25065024 IC50 = 7.6 nM T65200 C8GR2K 25065025 IC50 = 3.4 nM T65200 CEMG39 25065027 IC50 = 2.2 nM T65200 CB36SV 25065227 IC50 = 3.4 nM T65200 C7YH6J 25065230 IC50 = 3.4 nM T65200 C9EQ1D 25065231 IC50 = 8.9 nM T65200 CU12CJ 25065232 IC50 = 6.7 nM T65200 C8EVH3 25147627 IC50 = 40 nM T65200 CSQ5B7 25164121 IC50 = 5 nM T65200 CGW21A 25164133 IC50 = 14 nM T65200 CUT6A8 25181744 IC50 = 40 nM T65200 C4PJ6V 25182139 IC50 = 50 nM T65200 CRUF86 25182275 IC50 = 0.8 nM T65200 CS8R0I 25182553 IC50 = 4.4 nM T65200 C8O5VH 25182558 IC50 = 631 nM T65200 C9GFQ4 25183173 IC50 = 229 nM T65200 CZJ3G8 25183174 IC50 = 805 nM T65200 C2BI9A 25183175 IC50 = 64 nM T65200 CD7U6C 25183312 IC50 = 23 nM T65200 CHB16F 25183313 IC50 = 103 nM T65200 CTJZ86 25183314 IC50 = 42 nM T65200 CHYJ25 25183315 IC50 = 160 nM T65200 CZ27KB 25183604 IC50 = 29 nM T65200 C7V9UF 25183753 IC50 = 1.6 nM T65200 CUGV82 25192456 IC50 = 307 nM T65200 CCB2I0 25192603 IC50 = 110 nM T65200 CWRU15 25192607 IC50 = 12 nM T65200 CW09XG 25192736 IC50 = 3 nM T65200 CX5OM2 25192737 IC50 = 43 nM T65200 C06HNO 25192870 IC50 = 20 nM T65200 CXS91P 25192871 IC50 = 113 nM T65200 CI95ML 25192959 IC50 = 0.11 nM T65200 CL0YH1 25192961 IC50 = 3.3 nM T65200 CU0SD8 25192962 IC50 = 16.1 nM T65200 C4RQ5V 25192963 IC50 = 11.3 nM T65200 C5DI0O 25192964 IC50 = 361 nM T65200 CTRN65 25192965 IC50 = 4402 nM T65200 CRZ0X6 25193005 IC50 = 58 nM T65200 CY50LI 25193006 IC50 = 97 nM T65200 C9E6WR 25193007 IC50 = 76 nM T65200 C0J7LM 25193008 IC50 = 68 nM T65200 C5I0KR 25193009 IC50 = 994 nM T65200 C7R1CT 25193100 IC50 = 75 nM T65200 CVFK75 25193101 IC50 = 118 nM T65200 C36XRV 25193102 IC50 = 40 nM T65200 CA0MX2 25193144 IC50 = 178 nM T65200 C74NJG 25193145 IC50 = 124 nM T65200 CWU2E8 25193146 IC50 = 358 nM T65200 CEQF65 25210659 Ki = 12 nM T65200 CU09OD 25236186 IC50 = 4100 nM T65200 CW05JG 25263220 IC50 = 0.6 nM T65200 C05USX 25263221 IC50 = 3.8 nM T65200 C2K9FR 25263222 IC50 = 1.7 nM T65200 CZ0TK4 25263223 IC50 = 14 nM T65200 CU7E9B 25265683 IC50 = 10 nM T65200 C7BO2J 26009991 IC50 = 2631 nM T65200 CT10FO 32648983 IC50 = 13000 nM T65200 CPD4Z0 32684364 IC50 = 14490 nM T65200 CNK7V1 35856600 IC50 = 7200 nM T65200 CMRF64 36054265 IC50 = 20000 nM T65200 CP7RN3 36054272 IC50 > 100000 nM T65200 CSG4N6 36054289 IC50 = 15000 nM T65200 CQ65EV 36054707 IC50 = 12000 nM T65200 C3VML1 37529533 IC50 = 2106 nM T65200 CNI30Z 42603003 IC50 = 360 nM T65200 CMVE89 42603038 IC50 = 50 nM T65200 C79BRV 42603039 IC50 = 370 nM T65200 C1KU9S 42603075 IC50 = 25 nM T65200 C04TRI 42603076 IC50 = 4 nM T65200 CE0G6W 42633574 IC50 = 1280 nM T65200 CYC3O1 42634126 IC50 = 71 nM T65200 CK79IO 42634797 IC50 = 11 nM T65200 C9R7PZ 42634800 IC50 = 17 nM T65200 CX7D8M 42634801 IC50 = 5.9 nM T65200 CID91J 42634802 IC50 = 43 nM T65200 CH7ER1 42905087 IC50 = 36000 nM T65200 CW52HS 42906186 IC50 = 7300 nM T65200 CG82JI 42907599 IC50 = 7700 nM T65200 C7PO8U 42908115 IC50 = 64000 nM T65200 C94ESM 42915305 IC50 = 7300 nM T65200 CJE9Y6 42918799 IC50 = 53000 nM T65200 CI23FV 42921990 IC50 = 2100 nM T65200 CR0Y4M 42921991 IC50 = 20000 nM T65200 C8M3PB 42921992 IC50 = 10000 nM T65200 C17HTP 42921995 IC50 = 846 nM T65200 C5M7VH 44143287 IC50 = 2500 nM T65200 CTOD52 44143288 IC50 = 94 nM T65200 C6VQM9 44143289 IC50 = 25 nM T65200 C1FBL2 44143290 IC50 = 2100 nM T65200 CZ58CY 44143291 IC50 = 22 nM T65200 C8X2ZV 44143292 IC50 = 6 nM T65200 C6Q8TB 44143293 IC50 = 3 nM T65200 CKL98N 44143294 IC50 = 1410 nM T65200 CTHD32 44143295 IC50 = 445 nM T65200 CA32UQ 44143296 IC50 = 92 nM T65200 CE5VQ2 44143297 IC50 = 252 nM T65200 CV7B8I 44143298 IC50 = 1.5 nM T65200 C1IA7U 44143299 IC50 = 0.5 nM T65200 CNR9J0 44143306 Ki = 169 nM T65200 C5X2HM 44143308 Ki = 20 nM T65200 CL27SM 44143309 Ki = 5.8 nM T65200 C8KI3Z 44143310 Ki = 62 nM T65200 CQK48C 44143311 Ki = 4 nM T65200 CLA78S 44143312 Ki = 6.6 nM T65200 C96JKX 44143313 Ki = 1.9 nM T65200 CB46KU 44143314 Ki = 1.7 nM T65200 CIV01A 44143315 Ki = 9.8 nM T65200 CO2G0S 44155541 IC50 = 50 nM T65200 CD4N7Z 44155649 IC50 = 5 nM T65200 C65VWT 44155756 IC50 = 6 nM T65200 C63STN 44196869 IC50 = 25 nM T65200 C7YTM0 44197230 IC50 = 5.4 nM T65200 CKR4I6 44208369 IC50 = 31 nM T65200 COME74 44231030 IC50 = 353 nM T65200 CM8LV3 44231031 IC50 = 999 nM T65200 CK1Y3M 44236983 IC50 = 46 nM T65200 CV40JL 44237001 IC50 = 17 nM T65200 COZ3S8 44237012 IC50 = 45 nM T65200 C2XLK7 44237013 IC50 = 550 nM T65200 CPI5M8 44237014 IC50 = 20 nM T65200 C5XZJ7 44237015 IC50 = 18 nM T65200 C3E5KY 44237016 IC50 = 16 nM T65200 C6R4AH 44237017 IC50 = 15 nM T65200 CJHG60 44237018 IC50 = 667 nM T65200 CBS91O 44237019 IC50 = 14 nM T65200 C16AHN 44237020 IC50 = 922 nM T65200 C0O7AB 44237021 IC50 = 50 nM T65200 C0LZ4U 44237022 IC50 = 74 nM T65200 CF10AO 44237023 IC50 = 13 nM T65200 CIF5Z4 44237024 IC50 = 55 nM T65200 CHC0Y9 44237025 IC50 = 64 nM T65200 C8F4XE 44237026 IC50 = 7 nM T65200 CF0I5H 44237029 IC50 = 15 nM T65200 C5HY1I 44237030 IC50 = 390 nM T65200 CF48KO 44237031 IC50 = 9 nM T65200 C4A6MB 44237032 IC50 = 17 nM T65200 CTY7E8 44237033 IC50 = 58 nM T65200 CP7A0E 44237034 IC50 = 638 nM T65200 C05KHJ 44237035 IC50 = 11 nM T65200 C1MN8G 44237036 IC50 = 9 nM T65200 C6P5IL 44237037 IC50 = 29 nM T65200 CO32MH 44247592 IC50 = 9 nM T65200 CM54SL 44247841 IC50 = 15 nM T65200 CLBI82 44247842 IC50 = 97 nM T65200 CW3YT4 44247843 IC50 = 15 nM T65200 CX2HT8 44247844 IC50 = 10 nM T65200 CC70NL 44247845 IC50 = 10 nM T65200 CI04QP 44247973 IC50 = 136 nM T65200 CNA4H6 44247974 IC50 = 10 nM T65200 C3D0PI 44247975 IC50 = 40 nM T65200 CXM78K 44247976 IC50 = 18 nM T65200 C76JPE 44247977 IC50 = 63 nM T65200 CB0E6X 44248091 IC50 = 92 nM T65200 CHON16 44248092 IC50 = 10 nM T65200 CM2O6Y 44248093 IC50 = 200 nM T65200 CC70SD 44248094 IC50 = 100 nM T65200 C3WAR7 44248095 IC50 = 630 nM T65200 C3NYB1 44248096 IC50 = 10 nM T65200 C1WZT5 44248207 IC50 = 115 nM T65200 C3HZT2 44248208 IC50 = 11 nM T65200 C87VEH 44248209 IC50 = 50 nM T65200 C1X8FH 44248210 IC50 = 74 nM T65200 C8XT1A 44248211 IC50 = 10 nM T65200 C0D9WJ 44248333 IC50 = 17 nM T65200 CH63AC 44248334 IC50 = 11 nM T65200 CU0A2F 44248335 IC50 = 185000 nM T65200 CYRO42 44248336 IC50 = 639 nM T65200 CWH2Q4 44248337 IC50 = 10 nM T65200 C7T5XR 44248453 IC50 = 10 nM T65200 CO38EI 44248454 IC50 = 50 nM T65200 C8K7TJ 44248455 IC50 = 18 nM T65200 CW2Y5R 44248456 IC50 = 31 nM T65200 C6SVG1 44248577 IC50 = 674 nM T65200 CL6T9U 44248578 IC50 = 16 nM T65200 C9P6QL 44248579 IC50 = 28 nM T65200 C7M6WC 44248580 IC50 = 20 nM T65200 CC3V1W 44249656 IC50 = 190 nM T65200 CHA7J4 44250316 IC50 = 2 nM T65200 C4YE8N 44250392 IC50 = 56 nM T65200 C7UWV6 44251751 IC50 = 9 nM T65200 C2YQ5J 44251891 IC50 = 4 nM T65200 C2W6OE 44251893 IC50 = 4 nM T65200 CXEL39 44252043 IC50 = 28 nM T65200 C9UC3P 44252190 IC50 = 36 nM T65200 CMB0K6 44252191 IC50 = 30 nM T65200 C0PM5I 44252338 IC50 = 80 nM T65200 C2V3UY 44252339 IC50 = 68 nM T65200 CQ9GL3 44252340 IC50 = 60 nM T65200 CL1JV3 44252776 IC50 = 74 nM T65200 CL6XF7 44253232 IC50 = 31 nM T65200 CB97SH 44253510 IC50 = 54 nM T65200 CHV16X 44253783 IC50 = 395 nM T65200 C8ZC1O 44253785 IC50 = 27 nM T65200 C5C7XB 44253917 IC50 = 5670 nM T65200 CQJ73U 44253918 IC50 > 8000 nM T65200 C2V8UR 44253919 IC50 = 3180 nM T65200 C5LW8D 44253922 IC50 = 11 nM T65200 C8E1LF 44253923 IC50 = 10 nM T65200 CU8KV4 44402330 IC50 > 100000 nM T65200 C9S2HX 44402393 IC50 = 22908.68 nM T65200 CC0XN2 44402437 IC50 = 58700 nM T65200 C8C2QJ 44402534 IC50 = 17300 nM T65200 CW7IP2 44402550 IC50 = 47863.01 nM T65200 CWK8R1 44402659 IC50 > 100000 nM T65200 C0NUI2 44402662 IC50 = 100000 nM T65200 CM7LW8 44405286 IC50 = 22 nM T65200 CD13UE 44405324 IC50 = 2.57 nM T65200 CB42WK 44405337 IC50 = 9.3 nM T65200 CG45DB 44405340 IC50 = 4.1 nM T65200 CCX8Y5 44405353 IC50 = 4.074 nM T65200 CVU89O 44405363 IC50 = 1.9 nM T65200 CSH37Y 44405367 IC50 = 1.4 nM T65200 CRG59L 44405370 IC50 = 4.169 nM T65200 C4EK7T 44405379 IC50 = 7.2 nM T65200 C2GDM9 44405381 IC50 = 2 nM T65200 C75GUD 44405390 IC50 = 5.3 nM T65200 CHB1Z7 44405391 IC50 = 4.7 nM T65200 C9VQ6H 44405394 IC50 = 19.95 nM T65200 CQX58V 44405424 IC50 = 9.772 nM T65200 CLB4M5 44405433 IC50 = 4.898 nM T65200 C42FXZ 44418375 IC50 = 11 nM T65200 CC93VQ 44418376 IC50 = 80 nM T65200 CP9DO4 44418378 IC50 = 45 nM T65200 CR7K6S 44418382 IC50 = 5.012 nM T65200 C7B6GT 44418383 IC50 = 25.12 nM T65200 C1Q8CH 44418384 IC50 = 41 nM T65200 C7JNH9 44418385 IC50 = 89 nM T65200 CB58SX 44418389 IC50 = 15 nM T65200 CGKR51 44418390 IC50 = 6 nM T65200 CQT37N 44418391 IC50 = 28 nM T65200 CED27U 44418395 IC50 = 444 nM T65200 C9L7BU 44418396 IC50 = 185 nM T65200 C28DBM 44418400 IC50 = 5 nM T65200 C1KD8E 44418401 IC50 = 14 nM T65200 CT79UX 44418408 IC50 = 169 nM T65200 C7RW1O 44418409 IC50 = 29 nM T65200 C7WQD4 44418433 IC50 = 66 nM T65200 CV87RE 44418434 IC50 = 24 nM T65200 CE5W0V 44418440 IC50 = 269 nM T65200 CK74ZJ 44418441 IC50 = 75 nM T65200 C02AMZ 44418445 IC50 = 61.66 nM T65200 C7YCN4 44418447 IC50 = 306 nM T65200 C7AKJ2 44418450 IC50 = 43.65 nM T65200 C90QWN 44418451 IC50 = 35 nM T65200 CA2J1I 44418452 IC50 = 110 nM T65200 CE1W9Y 44418456 IC50 = 23 nM T65200 C7R3AT 44418457 IC50 = 637 nM T65200 C4MVN6 44418458 IC50 = 31 nM T65200 CXFR60 44418459 IC50 = 124 nM T65200 CC5Y6O 44418463 IC50 = 587 nM T65200 CAW7Z2 44418817 Ki = 180 nM T65200 C94IBD 44418818 Ki = 6 nM T65200 C97UNO 44418819 Ki = 6 nM T65200 CK90JF 44418820 Ki = 12 nM T65200 CC8ZR0 44418821 Ki = 3 nM T65200 CKX95Y 44418852 Ki = 21 nM T65200 CF56NG 44418856 Ki = 5 nM T65200 CGX84K 44418857 Ki = 4 nM T65200 CJ6V8K 44418859 Ki = 4 nM T65200 CSP8W1 44419286 IC50 = 35 nM T65200 CQH6X0 44419304 IC50 = 15 nM T65200 CBI64W 44419309 IC50 = 19 nM T65200 C6LOU9 44419313 IC50 = 230 nM T65200 C4IK2P 44419337 IC50 = 85 nM T65200 CKO36E 44419341 IC50 = 49 nM T65200 C32WUT 44420153 Ki = 8 nM T65200 C14JQE 44420164 Ki = 10 nM T65200 C76RGZ 44420166 Ki = 4 nM T65200 CINJ57 44420180 Ki = 16 nM T65200 CWM5F9 44420181 Ki = 53 nM T65200 CLA82E 44420186 Ki = 14 nM T65200 C0ET3O 44420190 Ki = 28 nM T65200 C3JF5Z 44420196 Ki = 17 nM T65200 C64UQO 44420202 Ki = 20 nM T65200 CJI76N 44420207 Ki = 60 nM T65200 C0T6ML 44420212 Ki = 700 nM T65200 C5Y4UB 44420215 Ki = 130 nM T65200 C1NCR3 44420232 Ki = 100 nM T65200 CQ7B8C 44420233 Ki = 13 nM T65200 C0X3PE 44420237 Ki = 10 nM T65200 CO4S5M 44420238 Ki = 19 nM T65200 CV6P7Y 44420242 Ki = 15 nM T65200 C8IH5C 44420243 Ki = 13 nM T65200 CZG60J 44420244 IC50 = 29 nM T65200 CN2B1J 44420246 Ki = 12 nM T65200 CG90VX 44420247 Ki = 22 nM T65200 C5PU7K 44420248 IC50 = 870 nM T65200 C7KW0L 44420249 Ki = 73 nM T65200 CBL6K2 44420251 IC50 = 36 nM T65200 CF9N4T 44420252 IC50 > 10000 nM T65200 CVX2Z3 44420253 Ki = 5 nM T65200 CX8IQ0 44420257 IC50 = 550 nM T65200 CN3W4S 44420259 Ki = 13 nM T65200 C1YLR4 44420285 Ki = 120 nM T65200 CNRY91 44420288 Ki = 560 nM T65200 CF23SE 44420291 Ki = 1100 nM T65200 CE7T4W 44420294 Ki = 22 nM T65200 CZRD26 44437603 IC50 = 4400 nM T65200 CP05CX 44437608 IC50 = 9300 nM T65200 CC1V7X 44437616 IC50 = 5000 nM T65200 CC3AW7 44437621 IC50 = 525 nM T65200 CBEV72 44437624 IC50 = 134 nM T65200 C4DZN7 44437625 IC50 = 169 nM T65200 CXZ87T 44437633 IC50 = 24000 nM T65200 C5F8TI 44437634 IC50 = 25000 nM T65200 CC63KF 44437635 IC50 > 100000 nM T65200 C91LMF 44437666 IC50 = 100000 nM T65200 CJ1O7N 44438556 IC50 = 38.9 nM T65200 CH0K4M 44438559 IC50 = 15 nM T65200 CXM65L 44438562 IC50 = 16 nM T65200 CM01KY 44438566 IC50 = 120 nM T65200 CFLP12 44438567 IC50 = 13 nM T65200 CAW10E 44438568 IC50 = 8.913 nM T65200 C3IK2C 44438569 IC50 = 110 nM T65200 C43RLG 44438570 IC50 = 96 nM T65200 CJX5B2 44438571 IC50 = 500 nM T65200 CM1Y7N 44438669 Ki = 26 nM T65200 CUE3I1 44438670 Ki = 8 nM T65200 CQM10L 44438671 Ki = 110 nM T65200 CB19EU 44438672 Ki = 5 nM T65200 CL4Y3J 44438673 Ki = 8 nM T65200 C7ON6I 44438675 Ki = 7 nM T65200 C5LN8W 44438676 Ki = 7 nM T65200 C8VI7M 44438677 Ki = 20 nM T65200 CV12KJ 44438678 Ki = 11 nM T65200 CBX9L4 44438679 Ki = 21 nM T65200 CP46XZ 44438680 Ki = 170 nM T65200 CF5YU4 44438681 Ki = 8 nM T65200 CJ2M3L 44438682 Ki = 3 nM T65200 CGM0A4 44440172 IC50 = 12000 nM T65200 CRJG19 44440202 IC50 = 24000 nM T65200 CQ7E2H 44440203 IC50 = 2100 nM T65200 C52HTK 44440204 IC50 = 8100 nM T65200 C1Z0YI 44440205 IC50 = 498 nM T65200 CL0Y2F 44443433 Ki > 10000 nM T65200 CWU53P 44443434 Ki = 450 nM T65200 CJB5H3 44443435 Ki = 110 nM T65200 C8RTU4 44443436 Ki = 180 nM T65200 CT26JD 44443437 Ki = 500 nM T65200 CQ1LB5 44443438 Ki = 1100 nM T65200 CT92KI 44443439 Ki = 1100 nM T65200 CZ1S4Y 44443440 Ki = 1600 nM T65200 C51UZM 44443441 Ki = 1700 nM T65200 CPG61T 44443442 Ki = 1300 nM T65200 C3U8IH 44443443 Ki = 270 nM T65200 C0JXQ9 44443444 Ki = 240 nM T65200 CP89WL 44443445 Ki = 170 nM T65200 CG96CE 44443446 Ki = 140 nM T65200 CKO16N 44443447 Ki = 330 nM T65200 C87NAF 44443448 Ki = 200 nM T65200 C6XHB1 44443449 Ki = 500 nM T65200 C9EV4Y 44443450 Ki = 180 nM T65200 CR5QC4 44443451 Ki = 360 nM T65200 C0ENK8 44448313 IC50 = 21 nM T65200 C7V5ET 44448422 IC50 = 1.9 nM T65200 CXG5Z9 44448462 IC50 = 2.7 nM T65200 CM97BK 44448463 IC50 = 1.4 nM T65200 C5V8HQ 44448464 IC50 = 9 nM T65200 CRW67T 44448507 IC50 = 26 nM T65200 C9RTN7 44448541 IC50 = 963 nM T65200 CRM3O9 44448543 IC50 = 12 nM T65200 C6HKY9 44448580 IC50 = 38 nM T65200 CK7BH0 44448581 IC50 = 50 nM T65200 C4NTZ7 44448583 IC50 = 13 nM T65200 CA2X5E 44448619 IC50 = 7.7 nM T65200 C6TDX0 44448620 IC50 = 260 nM T65200 CX4M7I 44448621 IC50 = 250 nM T65200 CJK8Y4 44448649 IC50 < 1 nM T65200 CM43XY 44448651 IC50 = 34 nM T65200 CI4Q9F 44448652 IC50 = 28 nM T65200 CADP58 44448655 IC50 = 28 nM T65200 CAP86X 44448671 IC50 = 89 nM T65200 CF0VR9 44448672 IC50 = 200 nM T65200 C56YZT 44448673 IC50 = 630 nM T65200 CG2O9U 44448674 IC50 = 90 nM T65200 CKC7P5 44448687 IC50 = 43 nM T65200 CX4J3Z 44448688 IC50 = 27 nM T65200 CMI0Y7 44448689 IC50 = 32 nM T65200 C08OCF 44448690 IC50 = 88 nM T65200 CK89RG 44448711 IC50 = 15 nM T65200 CU07RD 44448713 IC50 = 20 nM T65200 C5XV2W 44448731 IC50 = 3.6 nM T65200 C3U1WZ 44448872 IC50 = 35 nM T65200 C47YZF 44453649 IC50 = 52.48 nM T65200 C7CNI5 44453688 IC50 = 38.9 nM T65200 CDB14F 44453723 IC50 = 10.96 nM T65200 C9X8MG 44453874 IC50 = 4.677 nM T65200 CP8LS0 44453875 IC50 = 5.248 nM T65200 CN5Q7A 44453917 IC50 = 186.21 nM T65200 CR91NT 44453919 IC50 = 9.333 nM T65200 C6C0AZ 44453920 IC50 = 21.88 nM T65200 C8FLD9 44453964 IC50 = 181.97 nM T65200 CA6IQ1 44453966 IC50 = 28.18 nM T65200 CV1LI3 44453989 IC50 = 380.19 nM T65200 CKW73A 44453990 IC50 = 10 nM T65200 CCO39L 44453992 IC50 = 72.44 nM T65200 C1OH6E 44453993 IC50 = 5.012 nM T65200 CI3H8X 44454013 IC50 = 34.67 nM T65200 CW01YL 44454014 IC50 = 10.96 nM T65200 C6UDM8 44473368 IC50 = 12 nM T65200 CR2HV1 44473369 IC50 = 6.4 nM T65200 CA5UG3 44473378 IC50 = 5.4 nM T65200 CZ4MU8 44473379 IC50 = 66.9 nM T65200 CY7CI4 44473382 IC50 = 5.2 nM T65200 CX9TJ4 44476890 IC50 = 3.3 nM T65200 CUA9F0 44512094 IC50 = 1 nM T65200 C2T6KW 44561552 IC50 = 3800 nM T65200 CU9J5W 44564565 IC50 = 7.9 nM T65200 CJSW16 44564833 IC50 = 5.8 nM T65200 C3AZ1P 44564834 IC50 = 4.2 nM T65200 CZ92VC 44564876 IC50 = 2.2 nM T65200 CV5R6C 44564877 IC50 = 94 nM T65200 CGN54U 44564878 IC50 = 78 nM T65200 CTS3Y1 44564879 IC50 = 5 nM T65200 C7M5JR 44564921 IC50 = 36 nM T65200 C27DPG 44564922 IC50 = 96 nM T65200 C4EX9L 44564923 IC50 = 5.3 nM T65200 CP47LX 44564924 IC50 = 1 nM T65200 CJR2W9 44564925 IC50 = 11.3 nM T65200 CKYO28 44564974 IC50 = 4 nM T65200 C29WVL 44564975 IC50 = 70 nM T65200 CHWM49 44564976 IC50 = 16 nM T65200 CNL07P 44564977 IC50 = 30 nM T65200 C34RBP 44565028 IC50 = 55 nM T65200 C6O3ZB 44565029 IC50 = 8 nM T65200 CS1K2J 44565030 IC50 = 1.3 nM T65200 C26IDM 44565031 IC50 = 10 nM T65200 CN4Y9B 44565130 IC50 = 0.6 nM T65200 C2IH7W 44565131 IC50 = 0.8 nM T65200 C6UNO7 44565132 IC50 = 0.6 nM T65200 CO8UR7 44568341 IC50 = 370 nM T65200 CPC73X 44568372 IC50 = 1600 nM T65200 CAX16M 44568485 IC50 = 330 nM T65200 CJ97EW 44568578 IC50 = 69 nM T65200 CZ5A6G 44576636 IC50 = 1 nM T65200 CHD6G5 44576637 IC50 = 2.2 nM T65200 CK67LT 44576651 IC50 = 1.5 nM T65200 C9JB2Y 44576672 IC50 = 3.8 nM T65200 CMJ91U 44576707 IC50 = 10 nM T65200 C8D1LU 44576749 IC50 = 4.3 nM T65200 CKH1A8 44576750 IC50 = 11 nM T65200 CN93WV 44576751 IC50 = 68 nM T65200 CAH82I 44576752 IC50 = 14 nM T65200 CK5S4W 44576802 IC50 = 26 nM T65200 C9L3CP 44576803 IC50 = 3.5 nM T65200 C2F5RM 44576804 IC50 = 3 nM T65200 CK41XQ 44576805 IC50 = 44 nM T65200 CO5YU9 44576846 IC50 = 1 nM T65200 CH0X2J 44576847 IC50 = 12 nM T65200 CV6I1C 44576848 IC50 = 1 nM T65200 C9TC4U 44576849 IC50 = 11 nM T65200 C6ZU1A 44576872 IC50 = 1 nM T65200 C4YIR7 44576873 IC50 = 1.7 nM T65200 CRA54F 44576874 IC50 = 1 nM T65200 C2HW0I 44576875 IC50 = 0.98 nM T65200 C51WSL 44576899 IC50 = 2.6 nM T65200 CT62EL 44576900 IC50 = 6.9 nM T65200 CF2B1H 44576901 IC50 = 9.8 nM T65200 C0JH2G 44576902 IC50 = 0.98 nM T65200 C5M6GO 44576942 IC50 = 3.9 nM T65200 CWRD09 44576943 IC50 = 14 nM T65200 CWX1Z0 44576944 IC50 = 2.1 nM T65200 COQ7U4 44576945 IC50 = 0.98 nM T65200 C6P5ER 44576967 IC50 = 0.98 nM T65200 CED5X6 44583233 EC50 = 846 nM T65200 CX9S7W 44588424 IC50 = 14 nM T65200 C0N6DO 44625908 IC50 = 0.6 nM T65200 CXD90A 44625911 IC50 = 0.8 nM T65200 CV57ON 44814425 IC50 = 25 nM T65200 CSGN18 45268079 IC50 = 19 nM T65200 C18JAM 45269430 IC50 = 14 nM T65200 C97RUY 45269801 IC50 = 1200 nM T65200 CP5C8F 45270340 IC50 = 1130 nM T65200 CGPF36 45270351 IC50 = 49 nM T65200 C83OJH 45271081 IC50 = 47 nM T65200 C7O3DH 45271171 IC50 = 638 nM T65200 CH7X8N 45272362 IC50 > 1000 nM T65200 C6M1XW 45272365 IC50 > 1000 nM T65200 CE07FS 45272366 IC50 = 8 nM T65200 CTDH29 45272896 IC50 = 2698 nM T65200 C6WPN2 45272909 IC50 = 8512 nM T65200 CD57GF 45273834 IC50 = 411 nM T65200 CNS51G 46181099 IC50 = 46 nM T65200 CK65BP 46213656 IC50 = 1.1 nM T65200 CHI5S0 46216688 IC50 = 2 nM T65200 CAX31B 46216689 IC50 = 1.6 nM T65200 CN39HK 46229717 IC50 = 1508 nM T65200 C4VZD0 46230565 IC50 = 547 nM T65200 C56XLU 46230604 IC50 = 234 nM T65200 CMA96V 46230640 IC50 = 740 nM T65200 CI9Y0G 46230746 IC50 = 31 nM T65200 CWN85I 46230747 IC50 = 40 nM T65200 CU5OX3 46230748 IC50 = 720 nM T65200 CC1V3W 46231390 IC50 = 1.4 nM T65200 CK45RJ 46231437 IC50 = 0.9 nM T65200 CXZ6O9 46231438 IC50 = 1.1 nM T65200 CBJ4C7 46231439 IC50 = 2.2 nM T65200 C73FCP 46231440 IC50 = 0.8 nM T65200 C2W1ZY 46231441 IC50 = 0.9 nM T65200 CC4P1N 46231489 IC50 = 0.7 nM T65200 C9KW0X 46231490 IC50 = 41.6 nM T65200 CZ6N5X 46231491 IC50 = 56.8 nM T65200 C4N8DB 46231719 IC50 = 2 nM T65200 CF38WI 46231720 IC50 = 0.5 nM T65200 C4WT0Q 46231721 IC50 = 1.7 nM T65200 C0EG8P 46865563 IC50 = 1.4 nM T65200 C6ET9N 46880402 IC50 = 0.33 nM T65200 C06INV 46880490 IC50 = 547 nM T65200 C3U2CB 46880491 IC50 = 309 nM T65200 CMPE75 46880492 IC50 = 478 nM T65200 CC0VH7 46880554 IC50 = 137 nM T65200 C78SRI 46880555 IC50 = 1623 nM T65200 C4YJT6 46880556 IC50 = 740 nM T65200 CJ7B9Q 46880557 IC50 = 30 nM T65200 CZ0H3A 46880616 IC50 = 19 nM T65200 COSB92 46880617 IC50 = 32 nM T65200 CVT94J 46880618 IC50 = 48 nM T65200 C63UNR 46880662 IC50 = 114 nM T65200 CS79LH 46880663 IC50 = 159 nM T65200 CP6B4R 46880710 IC50 = 860 nM T65200 CR0J1C 46888800 Ki = 1.6 nM T65200 CZU6G3 46888801 IC50 = 0.03 nM T65200 COY09Z 46888802 IC50 = 0.03 nM T65200 C1O7YJ 46888803 IC50 = 0.32 nM T65200 C2J8ZS 46888840 IC50 = 0.32 nM T65200 CTA2M4 46888841 IC50 = 0.32 nM T65200 CXPO84 46888842 IC50 = 0.03 nM T65200 CC7J5N 46888843 IC50 = 0.32 nM T65200 CEJ48B 46888868 Ki = 1 nM T65200 CK6ZD0 46888869 Ki = 1 nM T65200 CW9FN6 46888870 IC50 = 0.34 nM T65200 C2G3BS 46888871 IC50 = 0.03 nM T65200 CY67QO 46889268 Ki = 15 nM T65200 C0FS3W 46889269 Ki = 2.4 nM T65200 C8J0KB 46890077 IC50 = 252 nM T65200 CHL91V 46890078 IC50 = 257 nM T65200 CTO16V 46890079 IC50 = 1300 nM T65200 C9N4YM 46890080 IC50 = 1340 nM T65200 C5ST1O 46890123 IC50 = 1050 nM T65200 CA50QX 46890124 IC50 = 1600 nM T65200 C37BWV 46890125 IC50 = 116 nM T65200 CT2M6N 46890126 IC50 = 289 nM T65200 CAO2J5 46890127 IC50 = 485 nM T65200 CJX5G0 46890128 IC50 = 1700 nM T65200 CK49GT 46890168 IC50 = 2180 nM T65200 CPCU19 46890169 IC50 = 954 nM T65200 C4LNV5 46890170 IC50 = 1660 nM T65200 CF6RA4 46890171 IC50 = 1450 nM T65200 CH4V3R 46890172 IC50 = 93 nM T65200 CNM31K 46890173 IC50 = 2450 nM T65200 COD69Y 46890203 IC50 = 1000 nM T65200 C3RVL0 46890204 IC50 = 1600 nM T65200 CECP45 46890205 IC50 = 1040 nM T65200 C46RBQ 46890206 IC50 = 860 nM T65200 CTL94D 46890207 IC50 = 1700 nM T65200 CU3MF2 46890241 IC50 = 1230 nM T65200 C2JC8G 46890242 IC50 = 943 nM T65200 C25TRJ 46890245 IC50 = 359 nM T65200 C5NTY2 46890246 IC50 = 2100 nM T65200 CDQ5H6 46890277 IC50 = 683 nM T65200 C9JE2A 46890278 IC50 = 948 nM T65200 CW2S6I 46890279 IC50 = 588 nM T65200 C4T6FY 46890280 IC50 = 114 nM T65200 C8SUK5 46890281 IC50 = 575 nM T65200 CRB2V3 46890282 IC50 = 2200 nM T65200 C7K2CB 46890308 IC50 = 304 nM T65200 C5L7VK 46890309 IC50 = 426 nM T65200 C2J3VX 46890310 IC50 = 686 nM T65200 C6B2OF 46890311 IC50 = 3900 nM T65200 CGI90V 46890312 IC50 = 1500 nM T65200 CVKI35 46890313 IC50 = 1100 nM T65200 C07GYC 46890334 IC50 = 8000 nM T65200 CHC48O 46890335 IC50 = 987 nM T65200 C24POT 46890336 IC50 = 915 nM T65200 CZ94OL 46890337 IC50 = 1500 nM T65200 C6AKF8 46890338 IC50 = 2400 nM T65200 CJ95DE 46890421 IC50 = 987 nM T65200 C64JBI 46890422 IC50 = 597 nM T65200 CVM9W2 46890423 IC50 = 4600 nM T65200 C4KX0O 46890424 IC50 = 310 nM T65200 CHW9O3 46890425 IC50 = 539 nM T65200 C0LIA9 46890426 IC50 = 215 nM T65200 CK0SX9 46890464 IC50 > 10000 nM T65200 C9E8RI 46890465 IC50 = 506 nM T65200 CN7J8E 46890466 IC50 = 843 nM T65200 CUBP32 46890467 IC50 = 751 nM T65200 C8FHZ2 46890468 IC50 = 493 nM T65200 C6RWK9 46890469 IC50 = 722 nM T65200 C5SYR1 46890513 IC50 = 1800 nM T65200 CM5JR0 46890514 IC50 = 1100 nM T65200 C0G9KB 46890515 IC50 > 10000 nM T65200 CBK06M 46890516 IC50 = 3900 nM T65200 C1R4PE 46890517 IC50 = 1900 nM T65200 C0OWJ3 46890518 IC50 = 4500 nM T65200 C93KGC 46890550 IC50 = 1100 nM T65200 CJL6S1 46890551 IC50 = 183 nM T65200 CIX36V 46894126 IC50 = 1010 nM T65200 CK9GS6 46906109 IC50 > 30000 nM T65200 CID25M 46906132 IC50 = 4650 nM T65200 CV79TC 46906133 IC50 = 12800 nM T65200 CX0G7D 46906134 IC50 = 4060 nM T65200 C1BUZ6 46906135 IC50 = 25600 nM T65200 C70MHI 46906136 IC50 = 3150 nM T65200 C9X0QR 46906171 IC50 = 7000 nM T65200 C1FWM3 46906172 IC50 > 30000 nM T65200 CN05UY 46906226 IC50 > 30000 nM T65200 C7UX2M 46906227 IC50 = 10600 nM T65200 CAB7O9 46906228 IC50 > 30000 nM T65200 CJ8NC4 46906252 IC50 = 3300 nM T65200 CU2C5J 46906253 IC50 > 30000 nM T65200 C6L2BD 46906254 IC50 = 5450 nM T65200 CFN1M5 46906255 IC50 = 9670 nM T65200 C8U1DE 46906280 IC50 = 3520 nM T65200 CB4P9Y 46906281 IC50 > 30000 nM T65200 CVXA62 46906282 IC50 = 4000 nM T65200 CDT8K7 46906283 IC50 = 6120 nM T65200 CZI7W2 46906284 IC50 = 6880 nM T65200 C2MJ7W 46906318 IC50 = 7000 nM T65200 CYD93Z 46906319 IC50 = 5930 nM T65200 CLCE52 46906320 IC50 = 23200 nM T65200 C31WXC 46906321 IC50 > 30000 nM T65200 CR1S9U 46906355 IC50 > 30000 nM T65200 C6QV3Z 46906356 IC50 = 23700 nM T65200 C5E8JV 46906357 IC50 > 30000 nM T65200 CY5M8V 46906378 IC50 = 18300 nM T65200 CKR18L 46906379 IC50 = 2790 nM T65200 CI96ZV 46906380 IC50 > 30000 nM T65200 C5QK2N 46906405 IC50 = 13500 nM T65200 CHZ13S 47006636 IC50 = 249 nM T65200 C28ULM 49713163 IC50 = 4800 nM T65200 CQWB45 49713168 IC50 = 18500 nM T65200 CS13YQ 49846481 IC50 = 10 nM T65200 CP5NT1 49846482 IC50 = 145 nM T65200 CSDQ25 49846544 IC50 = 20 nM T65200 CYVL63 49846545 IC50 = 50 nM T65200 CIS17B 49846687 IC50 = 10 nM T65200 CV3N2G 49846837 IC50 = 51 nM T65200 C6W2XQ 49846838 IC50 = 23 nM T65200 CJ8FU1 49846909 IC50 = 13 nM T65200 CIP23V 49846910 IC50 = 64 nM T65200 CE18TO 50925401 Ki = 143 nM T65200 C3Z5CA 50925402 Ki = 585 nM T65200 CC10UD 50994587 Ki = 173 nM T65200 CWE94G 50994588 Ki = 911 nM T65200 CC14RO 50994589 Ki = 585 nM T65200 CM2DP7 51186945 IC50 = 275 nM T65200 CL0QN8 52911312 IC50 = 20 nM T65200 CUD24Z 52911829 IC50 = 31 nM T65200 C6K8LB 52911830 IC50 = 23 nM T65200 C81QFB 52911831 IC50 = 38 nM T65200 C8TPV1 52911882 IC50 = 29 nM T65200 CH0LF9 52911883 IC50 = 27 nM T65200 CO8U3V 52911884 IC50 = 26 nM T65200 C5GK3T 52911885 IC50 = 22 nM T65200 C7C8ZG 52911886 IC50 = 22 nM T65200 CMJ09C 52911940 IC50 = 15 nM T65200 C16JFX 52911941 IC50 = 45 nM T65200 CFRZ03 52911942 IC50 = 94 nM T65200 C79ZAT 52911944 IC50 = 25 nM T65200 CA8N9P 52911994 IC50 = 1.6 nM T65200 CLE06Z 52912040 IC50 = 20 nM T65200 C2U1HZ 52912042 IC50 = 14 nM T65200 CI47YN 52912091 IC50 = 12 nM T65200 C89GXD 52912092 IC50 = 30 nM T65200 CH5X4A 52912093 IC50 = 48 nM T65200 CQF7S5 52912094 IC50 = 30 nM T65200 CG32UO 52912144 IC50 = 11 nM T65200 CICZ45 52918012 IC50 = 43 nM T65200 C4X2WF 52939227 IC50 > 40000 nM T65200 CQ6R0S 52939228 IC50 = 45000 nM T65200 CB9G7Y 52940874 IC50 = 15.7 nM T65200 C3QHN6 52940894 IC50 = 21.3 nM T65200 C10WZR 52940895 IC50 = 1.1 nM T65200 CU0J9O 52940907 IC50 = 14.7 nM T65200 C1YRT3 52940913 IC50 = 61.9 nM T65200 CSXY62 52941059 IC50 = 0.4 nM T65200 C1XY9O 52941171 IC50 = 4.7 nM T65200 C2WZN8 52941220 IC50 = 11 nM T65200 CXF8J2 52941221 IC50 = 1.2 nM T65200 CTQS02 52941278 IC50 = 50 nM T65200 C1JL4P 52941329 IC50 > 300 nM T65200 CS4C7A 52941374 IC50 = 3.2 nM T65200 CA07SN 52941527 IC50 = 125 nM T65200 C6NR7I 52942081 IC50 = 3.4 nM T65200 C3BO1Z 52942119 IC50 = 0.63 nM T65200 CM7KW2 52942143 IC50 = 68 nM T65200 C9OG8P 52942175 IC50 = 2 nM T65200 C1PAR9 52942397 IC50 = 36.6 nM T65200 C6SMK9 52942398 IC50 = 24 nM T65200 CG0DU9 52942765 IC50 = 36 nM T65200 C3TK2O 52943442 IC50 = 7.6 nM T65200 CPH49F 52943645 IC50 = 1.2 nM T65200 C8L2OX 52943755 IC50 = 2 nM T65200 C89JFD 52943843 IC50 = 110 nM T65200 C0OQ9H 52943893 IC50 = 14 nM T65200 CSRI98 52944465 IC50 = 17.6 nM T65200 CVE4J6 52944478 IC50 = 20.7 nM T65200 CX0YD9 52944600 IC50 = 5.2 nM T65200 CXTM57 52944645 IC50 = 2.7 nM T65200 C5GS6Z 52944762 IC50 = 79 nM T65200 C9OV7S 52945102 IC50 = 86 nM T65200 C3O4AU 52945262 IC50 = 4.1 nM T65200 C8X4NE 52945350 IC50 = 626 nM T65200 CT01CE 52945715 IC50 = 5.8 nM T65200 C3J2FA 52945716 IC50 = 98 nM T65200 CE3AQ9 52945888 IC50 = 825 nM T65200 CMED86 52946026 IC50 = 229 nM T65200 CZ4TI9 52946104 IC50 = 280 nM T65200 CVH40Q 52946155 IC50 = 109 nM T65200 CCD34R 52946156 IC50 = 144 nM T65200 C48WFA 52946320 IC50 = 184 nM T65200 CBV0Q9 52946391 IC50 = 0.6 nM T65200 C5SP8F 52946462 IC50 = 7.4 nM T65200 CL2T8B 52946549 IC50 = 289 nM T65200 C3LMK2 52946948 IC50 = 7 nM T65200 CO7ZR1 52947102 IC50 = 2.7 nM T65200 C2KHL7 52947144 IC50 = 42.7 nM T65200 C8WZY5 52947559 IC50 = 30 nM T65200 CS9C3I 52947617 IC50 = 0.9 nM T65200 C2YK4B 52947710 IC50 = 2.7 nM T65200 C1TW8M 52947732 IC50 > 300 nM T65200 CBE50I 52948127 IC50 = 15.3 nM T65200 C56NDZ 52948169 IC50 = 1.4 nM T65200 CNXJ68 52948209 IC50 = 2.9 nM T65200 C5MJG3 52948460 IC50 = 317 nM T65200 C43KTX 52948925 IC50 = 0.82 nM T65200 CC4E3P 52949552 IC50 = 20 nM T65200 CQ6D2J 52949732 IC50 = 7.5 nM T65200 C23DBP 52949843 IC50 = 1.8 nM T65200 C5MYL0 52949904 IC50 = 30 nM T65200 CUJ68Z 52950064 IC50 = 1.2 nM T65200 CJI28A 52950107 IC50 = 929 nM T65200 CZX96L 53316802 IC50 = 10 nM T65200 COU02M 53317315 IC50 = 2.4 nM T65200 CQ8D1F 53317316 IC50 = 554 nM T65200 CED72G 53317317 IC50 = 10 nM T65200 CH6E4Q 53317318 IC50 = 683 nM T65200 CME8T9 53317319 IC50 = 67 nM T65200 C56EHQ 53317320 IC50 = 11 nM T65200 C8BI6Z 53317725 IC50 = 2130 nM T65200 C3TSB5 53319921 IC50 = 24 nM T65200 C12JKN 53319922 IC50 = 10 nM T65200 CDF72K 53319923 IC50 = 8 nM T65200 CD86YE 53320073 IC50 = 10 nM T65200 CR64ZG 53320074 IC50 = 3 nM T65200 CV6I9H 53320291 IC50 = 8.8 nM T65200 CEHQ08 53320743 IC50 = 2 nM T65200 CA03EQ 53320744 IC50 = 20 nM T65200 CW4ZQ5 53321227 IC50 = 1.9 nM T65200 CZ3W1N 53321228 IC50 = 3.9 nM T65200 CR5I1K 53321229 IC50 = 17 nM T65200 CL2Q4A 53321230 IC50 = 170 nM T65200 CI1N3E 53322042 IC50 = 12 nM T65200 CJD3T7 53322558 IC50 = 16 nM T65200 CSUK37 53322740 IC50 = 8300 nM T65200 CQ7J8E 53322756 IC50 = 4000 nM T65200 C54BDO 53323882 IC50 = 0.6 nM T65200 CRD6K2 53323883 IC50 = 3.5 nM T65200 CNK20C 53323884 IC50 = 55 nM T65200 CP1LV4 53323885 IC50 = 149 nM T65200 CDT61L 53323886 IC50 = 10 nM T65200 CGVR94 53323887 IC50 = 5 nM T65200 CQ2XT9 53324358 IC50 = 5 nM T65200 C2EDQ5 53324718 IC50 = 37 nM T65200 C1P8HX 53325169 IC50 = 20 nM T65200 C8Z7QR 53325170 IC50 = 1.3 nM T65200 COZ3I5 53325171 IC50 = 63 nM T65200 C68PHG 53325172 IC50 = 945 nM T65200 CMHV08 53326462 IC50 = 9.6 nM T65200 CJ7Y2I 53326463 IC50 = 20 nM T65200 C9D4UK 53326464 IC50 = 20 nM T65200 CSU34Y 53326465 IC50 = 11 nM T65200 C6W3JM 53326660 IC50 = 5400 nM T65200 CP91BU 53326661 IC50 > 10000 nM T65200 CORJ01 53326800 IC50 = 16 nM T65200 C9H5YE 53361128 IC50 = 0.8 nM T65200 C08UFV 53470409 IC50 = 270 nM T65200 CL19HU 53473036 IC50 > 100 nM T65200 C9WZ3S 53473134 IC50 = 8.4 nM T65200 CE74YF 53473135 IC50 = 0.7 nM T65200 CO3W2B 53473136 IC50 = 0.5 nM T65200 C3SF8E 53473137 IC50 = 0.4 nM T65200 CPN3C9 53473138 IC50 = 18.7 nM T65200 CQNO62 53473139 IC50 = 2.1 nM T65200 C8L2MJ 53473230 IC50 = 1.2 nM T65200 CN1W0A 53473231 IC50 = 1.3 nM T65200 CY1DW7 53473232 IC50 = 14.7 nM T65200 CNS4A7 53473233 IC50 = 0.5 nM T65200 CCN3Q2 53473234 IC50 = 12 nM T65200 CL7D1V 53473235 IC50 = 2.7 nM T65200 C0VSY7 53473320 IC50 = 34 nM T65200 CZ8DA1 53473321 IC50 = 0.8 nM T65200 CU7OV5 53473322 IC50 = 16 nM T65200 C8J4VI 53473323 IC50 = 69 nM T65200 C1HPT4 53473324 IC50 = 1 nM T65200 CUN1Z2 53473393 IC50 = 11 nM T65200 CE0I2P 53473394 IC50 = 5 nM T65200 CEW1G6 53473395 IC50 = 22 nM T65200 CW3Q5H 53473396 IC50 = 5.7 nM T65200 CY0WF5 53473397 IC50 = 1.4 nM T65200 C79FHR 53473483 IC50 = 4.1 nM T65200 CS87DG 53473484 IC50 = 32 nM T65200 CW2ZK6 53474283 IC50 = 92 nM T65200 CO7N3X 53474284 IC50 > 100 nM T65200 C03WNH 53474286 IC50 = 50 nM T65200 CN93FS 54580118 IC50 = 1 nM T65200 CF05VK 54580143 IC50 = 120 nM T65200 C7FXV6 54580144 IC50 = 5.5 nM T65200 C2M8XQ 54580210 IC50 = 4 nM T65200 C4Q6MO 54580243 IC50 = 900 nM T65200 CQKX72 54580341 IC50 = 436 nM T65200 CLT8C3 54580342 IC50 = 93 nM T65200 C8QCX2 54580343 IC50 = 4 nM T65200 CR1S8I 54580344 IC50 = 37 nM T65200 CBX17R 54581094 IC50 = 540 nM T65200 C8O9WK 54581095 IC50 < 1 nM T65200 C8ZDF3 54581137 IC50 = 1.8 nM T65200 C14YRS 54581213 IC50 = 30 nM T65200 CU12AD 54581342 IC50 > 2000 nM T65200 CG5BI4 54581343 IC50 = 127 nM T65200 CM3TF1 54581344 IC50 = 18 nM T65200 CQ7GV2 54582134 IC50 = 300 nM T65200 CZ1B6L 54582135 IC50 = 250 nM T65200 CK29GC 54582137 IC50 = 1.5 nM T65200 CKGX19 54582164 IC50 = 2.2 nM T65200 CWA6Q0 54582242 IC50 < 1 nM T65200 C07LYE 54582261 IC50 = 8.1 nM T65200 CP2N1C 54582262 IC50 = 7.5 nM T65200 CT6UM8 54582370 IC50 = 40 nM T65200 CM2QX4 54583079 IC50 = 560 nM T65200 CMKQ26 54583080 IC50 < 1 nM T65200 C2G7LK 54583125 IC50 = 1.2 nM T65200 CL6Z9X 54583126 IC50 = 14 nM T65200 CGM2W4 54583127 IC50 = 4.8 nM T65200 CF42QY 54583128 IC50 = 4.8 nM T65200 CWHS39 54583210 IC50 = 2 nM T65200 CDK5V0 54583231 IC50 = 11 nM T65200 C5V4DY 54583232 IC50 = 4.4 nM T65200 C1JV9N 54583233 IC50 = 3.7 nM T65200 CKA9L3 54583234 IC50 = 2800 nM T65200 CM0KW4 54583345 IC50 > 2000 nM T65200 C3IP2G 54583346 IC50 > 2000 nM T65200 CU3C9Z 54583347 IC50 = 378 nM T65200 CIV10X 54583348 IC50 > 2000 nM T65200 CL8P1K 54583349 IC50 = 27 nM T65200 CP9L4D 54583350 IC50 = 7 nM T65200 CZ4YV3 54584081 IC50 = 470 nM T65200 CHP62C 54584119 IC50 = 2.3 nM T65200 CCT0B2 54584121 IC50 = 2.8 nM T65200 C0VPS6 54584122 IC50 = 3.7 nM T65200 C6P5XR 54584196 IC50 = 20 nM T65200 CY2WM3 54584197 IC50 = 4.1 nM T65200 CXNP26 54584198 IC50 = 20 nM T65200 CN71SQ 54584299 IC50 > 2000 nM T65200 CJ2E8S 54584300 IC50 = 9 nM T65200 CWY83C 54584415 IC50 = 5.5 nM T65200 CGD4N3 54585028 IC50 = 76 nM T65200 C8NZ2B 54585029 IC50 = 69 nM T65200 CHW48S 54585030 IC50 = 2.6 nM T65200 CZ8R0S 54585053 IC50 = 1.5 nM T65200 C04IZR 54585054 IC50 = 11 nM T65200 C6GZB9 54585157 IC50 = 140 nM T65200 C1T2BD 54585261 IC50 = 73 nM T65200 C5SHO2 54585992 IC50 = 5.8 nM T65200 CJA5Z6 54585993 IC50 = 69 nM T65200 C4JTZ5 54585994 IC50 = 8.7 nM T65200 CKF15E 54586030 IC50 = 2.2 nM T65200 CT12RX 54586031 IC50 = 1.1 nM T65200 CD6FC5 54586091 IC50 < 1 nM T65200 CDG95F 54586092 IC50 = 1 nM T65200 CMIQ74 54586218 IC50 = 100 nM T65200 CJ8K1Y 54586966 IC50 = 650 nM T65200 C51MDN 54586967 IC50 = 11 nM T65200 CH2F8P 54586968 IC50 = 9.5 nM T65200 C61ZTA 54586969 IC50 = 8 nM T65200 C3Y6HF 54587012 IC50 = 1.5 nM T65200 CUF68X 54587090 IC50 = 1.1 nM T65200 CI1PV5 54587121 IC50 = 3.3 nM T65200 C6PSJ3 54587122 IC50 = 5.1 nM T65200 C9D1UH 54587123 IC50 = 1.6 nM T65200 C82TDJ 54587124 IC50 = 10 nM T65200 CF2CG0 54587243 IC50 > 2000 nM T65200 CQ8BH1 54587244 IC50 = 8 nM T65200 C43SOJ 54587245 IC50 = 67 nM T65200 CM61OP 54590875 IC50 = 8.7 nM T65200 CNQ41E 54590876 IC50 = 3.9 nM T65200 CQ0R6D 54590877 IC50 = 5.5 nM T65200 CXE18A 54590878 IC50 = 4.3 nM T65200 CN73JM 54590965 IC50 = 2.3 nM T65200 CR3VL2 54590966 IC50 = 1.8 nM T65200 C39YQP 54591053 IC50 = 2.4 nM T65200 CK9TA7 54591214 IC50 = 2.7 nM T65200 C1PC3R 54591293 IC50 = 9.2 nM T65200 CHQ5G7 54591749 IC50 = 2.7 nM T65200 CD09KX 54591819 IC50 = 1.7 nM T65200 CACN12 54591821 IC50 = 3.9 nM T65200 C0YCF1 54591822 IC50 = 3.2 nM T65200 CFY71J 54591823 IC50 = 3.2 nM T65200 CY1Z6T 54591824 IC50 = 1.9 nM T65200 CE0SJ5 54591902 IC50 = 6.8 nM T65200 CSL97G 54591982 IC50 = 2.8 nM T65200 CV10QA 54591983 IC50 = 3.1 nM T65200 C3YI2S 54591984 IC50 = 9.5 nM T65200 CG6PQ3 54591985 IC50 = 3.4 nM T65200 CS29OJ 54592059 IC50 = 4.2 nM T65200 C79MTC 54592060 IC50 = 35 nM T65200 CY0S5T 54592061 IC50 = 2 nM T65200 COL0D8 54592062 IC50 = 2.1 nM T65200 CQC2E0 54679348 IC50 = 4500 nM T65200 CT62JH 54728117 IC50 = 3000 nM T65200 CO7HG2 54754506 IC50 = 34 nM T65200 CLXD72 54754620 IC50 = 1 nM T65200 CA6OM2 54754622 IC50 = 2 nM T65200 C8FA7C 54754623 IC50 = 1 nM T65200 CZTD58 54754864 IC50 = 190 nM T65200 CF4OW7 54754981 IC50 = 80 nM T65200 CZ5NP7 54755452 IC50 = 4 nM T65200 CZMB04 54755700 IC50 = 12 nM T65200 C37PTV 54755821 IC50 = 4 nM T65200 C5DO9M 54755941 IC50 = 54 nM T65200 CP7N5U 54756055 IC50 = 1 nM T65200 CB7RN0 54756059 IC50 = 2 nM T65200 CALV13 54756172 IC50 = 1 nM T65200 C5GRV8 54756173 IC50 = 2 nM T65200 CE63XU 54756287 IC50 = 1 nM T65200 CI4UF8 54756403 IC50 = 1 nM T65200 C6KY3N 54756407 IC50 = 1 nM T65200 C7A6ZL 56649596 IC50 = 1000 nM T65200 CDS9Y3 56659419 IC50 = 5.5 nM T65200 C6RU0N 56659420 IC50 = 5.6 nM T65200 C59BZL 56659421 IC50 = 367 nM T65200 C9T2UJ 56662869 IC50 = 544 nM T65200 CM4EH1 56662870 IC50 = 48240 nM T65200 CSNX08 56662871 IC50 = 64 nM T65200 CC4ME1 56666351 IC50 = 2.8 nM T65200 CCRD50 56666352 IC50 = 1298 nM T65200 CHAZ26 56666380 IC50 = 578 nM T65200 CB5P7A 56669762 IC50 = 7804 nM T65200 C2XBV7 56673255 IC50 = 197 nM T65200 CI54DZ 56676581 IC50 = 163 nM T65200 C9ASY6 56676582 IC50 = 939 nM T65200 CU27YF 56676583 IC50 = 16060 nM T65200 C7JC4S 56679928 IC50 = 8778 nM T65200 CF1O6J 56679929 IC50 = 8.2 nM T65200 C9O1JQ 56683245 IC50 = 17 nM T65200 CQ4H9K 56683246 IC50 = 3.7 nM T65200 C9VWL0 56683247 IC50 = 14030 nM T65200 C3NPO1 56683248 IC50 = 8.5 nM T65200 CC4K6F 56683271 IC50 = 36 nM T65200 C7C8UQ 57240144 IC50 = 694 nM T65200 CIO89K 57390996 IC50 = 135 nM T65200 CMR1N0 57390998 IC50 = 31 nM T65200 CFJ91L 57390999 IC50 = 93 nM T65200 C6BPL1 57392755 IC50 = 48 nM T65200 C1S0EA 57392783 IC50 = 4 nM T65200 C4V9LD 57392784 IC50 = 3 nM T65200 C3IAB0 57392785 IC50 = 5 nM T65200 CJKU19 57392786 IC50 = 8 nM T65200 C31VBE 57394414 IC50 = 127 nM T65200 CC9UZ0 57394415 IC50 = 240 nM T65200 C2CU5V 57394511 IC50 > 10 nM T65200 CCT90V 57396247 IC50 = 189 nM T65200 C1CUV9 57396248 IC50 = 425 nM T65200 C09MIU 57396256 IC50 = 12 nM T65200 C1KNY7 57396257 IC50 = 9 nM T65200 COZ0C4 57396258 IC50 = 3 nM T65200 C56VTZ 57396259 IC50 = 396 nM T65200 C43JML 57398049 IC50 = 14 nM T65200 C9J4VH 57398058 IC50 = 225 nM T65200 C3SD6C 57398060 IC50 = 11 nM T65200 C30WYE 57398061 IC50 = 13 nM T65200 C9NC0U 57398062 IC50 = 6 nM T65200 C7AJ4Q 57398139 IC50 = 7 nM T65200 CW9ZM6 57399703 IC50 = 153 nM T65200 CYMA01 57399704 IC50 = 2203 nM T65200 C0XQ8W 57399705 IC50 = 4705 nM T65200 C7EOG6 57399717 IC50 = 15 nM T65200 CSD28Q 57401469 IC50 = 234 nM T65200 CBFQ56 57401481 IC50 = 104 nM T65200 C4OG3X 57401482 IC50 = 8 nM T65200 CTI4L7 57401483 IC50 = 8 nM T65200 C3K5SY 57403224 IC50 = 269 nM T65200 C53KUF 57403225 IC50 = 4 nM T65200 CO49PY 57403226 IC50 = 10 nM T65200 C4CE1X 57403227 IC50 = 332 nM T65200 CAET30 57403315 IC50 = 49 nM T65200 CMD10R 57404453 EC50 = 517 nM T65200 C4I9DE 57408764 IC50 = 105 nM T65200 CM2DN9 57408765 IC50 = 72 nM T65200 C81NES 57418435 IC50 = 15 nM T65200 CAI0P1 57418438 IC50 = 17 nM T65200 CG2H5V 57418439 IC50 = 10 nM T65200 CAW03D 57576883 IC50 = 349 nM T65200 CC09EQ 57576892 IC50 = 1700 nM T65200 C1EC2O 57576905 IC50 = 308 nM T65200 CE18AC 57576921 IC50 = 3600 nM T65200 CXHJ84 57576960 IC50 = 655 nM T65200 C79HCK 57576967 IC50 = 165 nM T65200 C09DEG 57576970 IC50 = 448 nM T65200 C0G3FS 57576977 IC50 = 2200 nM T65200 C6S1MY 57576996 IC50 = 125 nM T65200 CWUR92 57577004 IC50 = 229 nM T65200 CCTP46 57577008 IC50 = 1080 nM T65200 CK91TC 57577024 IC50 = 2880 nM T65200 CN7YT4 57652306 IC50 = 0.5 nM T65200 CJ17LO 57808861 IC50 = 1 nM T65200 C3XQZ4 57808870 IC50 = 2.7 nM T65200 C0GN3C 57808912 IC50 = 0.5 nM T65200 CK3E2N 57808982 IC50 = 21 nM T65200 CL38KT 57808983 IC50 = 1.4 nM T65200 CRDS36 57808989 IC50 = 0.9 nM T65200 CDY2J9 57808991 IC50 = 5.1 nM T65200 C39YAD 57809000 IC50 = 0.7 nM T65200 C05XBJ 57809011 IC50 = 5.5 nM T65200 CCFD09 57809042 IC50 = 22 nM T65200 CQP0Z8 57916308 IC50 = 1200 nM T65200 C7KH3J 57916338 IC50 = 16 nM T65200 CSPK27 57916353 IC50 = 9 nM T65200 C39SNL 57916360 IC50 = 14 nM T65200 C8GY7X 57916364 IC50 = 23 nM T65200 CQXC05 57916383 IC50 = 94 nM T65200 C0WD4E 57916384 IC50 = 137 nM T65200 CXJ8R7 57916392 IC50 = 847 nM T65200 CMC52X 57916394 IC50 = 1480 nM T65200 C30LQO 57916397 IC50 = 108 nM T65200 C5F2XD 57916410 IC50 = 21 nM T65200 CKO2D5 57916411 IC50 = 644 nM T65200 C9X0OU 57916416 IC50 = 2100 nM T65200 CSJ18W 57916434 IC50 = 19 nM T65200 CIB78R 57916440 IC50 = 4.5 nM T65200 CU4OF3 57916448 IC50 = 46 nM T65200 C3I9VS 57916457 IC50 = 14800 nM T65200 C2JF0A 57916458 IC50 = 22 nM T65200 C6FHZ4 57916469 IC50 = 30 nM T65200 CD52SU 57916480 IC50 = 13 nM T65200 CWO82G 57916485 IC50 = 12 nM T65200 CG16CV 57916503 IC50 = 102 nM T65200 C21FSD 57916516 IC50 = 53 nM T65200 C64SHV 57941312 IC50 = 14 nM T65200 C9NQ0O 57941349 IC50 = 8 nM T65200 CR8T9F 57941389 IC50 = 9 nM T65200 CQVY45 57941391 IC50 = 89 nM T65200 CM14GC 57941400 IC50 = 31 nM T65200 CG23VP 57941404 IC50 = 13 nM T65200 CYM4N1 57941436 IC50 = 20 nM T65200 CR10NP 57941439 IC50 = 22 nM T65200 C69HUA 57941440 IC50 = 634 nM T65200 C20UHY 57941482 IC50 = 23 nM T65200 CE7MQ6 57941504 IC50 = 60 nM T65200 C1CM6O 57941506 IC50 > 22000 nM T65200 C6C8UT 57941522 IC50 = 31 nM T65200 CGV8Z6 58000867 IC50 = 32 nM T65200 CDXB56 58109207 IC50 = 10.6 nM T65200 CF06NM 58109212 IC50 = 0.7 nM T65200 CSC1K6 58109236 IC50 = 1 nM T65200 C2Q8AR 58109239 IC50 = 1.4 nM T65200 CS05MK 58109240 IC50 = 2.5 nM T65200 CDC28F 58109250 IC50 = 1.2 nM T65200 CY5V0J 58109251 IC50 = 0.8 nM T65200 CX3QK5 58109370 IC50 = 2.3 nM T65200 C4E2RC 58109371 IC50 = 0.8 nM T65200 C2EY8P 58109378 IC50 = 2 nM T65200 C5LUH2 58109381 IC50 = 80 nM T65200 CR62JC 58109389 IC50 = 14.5 nM T65200 C05LAK 58109398 IC50 = 2.3 nM T65200 C0ONJ3 58109407 IC50 = 2.2 nM T65200 C75ZBE 58109449 IC50 = 7.7 nM T65200 CJ07OW 58109450 IC50 = 1.1 nM T65200 C5JGU1 58109561 IC50 = 2 nM T65200 C0T4IE 58109574 IC50 = 4.1 nM T65200 CST59B 58109619 IC50 = 65.9 nM T65200 CZAJ57 58109626 IC50 = 1.7 nM T65200 CZY78L 58109663 IC50 = 1.2 nM T65200 CK8B6T 58109672 IC50 = 4.8 nM T65200 C4SC0Z 58109674 IC50 = 1.1 nM T65200 CNUV29 58109685 IC50 = 3.6 nM T65200 CTQ2N4 58109704 IC50 = 0.6 nM T65200 CRZU03 58109712 IC50 = 1.3 nM T65200 C4NJG2 58109725 IC50 = 0.7 nM T65200 C1EF0B 58109729 IC50 = 2.6 nM T65200 C6JXZ1 58210551 IC50 = 310 nM T65200 CO43YS 58210558 IC50 = 20 nM T65200 CG1K7Y 58210578 IC50 = 220 nM T65200 CWR8Y3 58210632 IC50 = 52 nM T65200 CIYE10 58210659 IC50 = 110 nM T65200 CDY78I 58210755 IC50 = 160 nM T65200 CD73AV 58210762 IC50 = 16000 nM T65200 CDRN63 58210800 IC50 = 5 nM T65200 CK96UZ 58210815 IC50 = 92 nM T65200 C8S9GL 58210850 IC50 = 11000 nM T65200 C5AIV8 58210920 IC50 = 21000 nM T65200 CRV1B8 58210955 IC50 = 120 nM T65200 CP1C3U 58210962 IC50 = 180 nM T65200 C0WDO1 58210998 IC50 = 49 nM T65200 CC51VS 58211029 IC50 = 1300 nM T65200 CA5XB4 58211042 IC50 = 430 nM T65200 CAZ5N9 58211074 IC50 = 3 nM T65200 CU2G7J 58211112 IC50 = 9 nM T65200 CV6D5F 58211134 IC50 = 5800 nM T65200 CG1SX3 58211235 IC50 = 18000 nM T65200 C4OBD1 58211257 IC50 = 26000 nM T65200 C7XVL3 58211263 IC50 = 720 nM T65200 CXTE12 58211270 IC50 = 220 nM T65200 C7OG1U 58211295 IC50 = 320 nM T65200 C08MJC 58211376 IC50 = 25000 nM T65200 CEY4H8 58211430 IC50 = 9 nM T65200 CZ7C3H 58211448 IC50 = 2600 nM T65200 CF5OX9 58211491 IC50 = 13000 nM T65200 C1GWK7 58211501 IC50 = 55 nM T65200 C3B9XP 58211552 IC50 = 320 nM T65200 CF5MR9 58211634 IC50 = 30 nM T65200 C1I5DU 58211666 IC50 = 980 nM T65200 C67JSA 58324675 IC50 = 22 nM T65200 CWYK20 58485289 IC50 = 0.5 nM T65200 CN2E9O 58485355 IC50 = 0.4 nM T65200 CQNG37 58485380 IC50 = 1.7 nM T65200 CVH1M2 58708330 IC50 = 300 nM T65200 CPN47R 58730567 IC50 = 180 nM T65200 CJ68WA 59336862 IC50 = 0.3 nM T65200 CJS6Y0 59336934 IC50 = 175 nM T65200 C5KOB7 59336970 IC50 = 12 nM T65200 CTVM01 59337052 IC50 = 2 nM T65200 CAV16J 59337131 IC50 = 63 nM T65200 CNG95D 59337133 IC50 = 3 nM T65200 CQ2V4T 59337171 IC50 = 17 nM T65200 C6G9ID 59337183 IC50 = 3 nM T65200 CGY7A1 59337189 IC50 = 8 nM T65200 C6E5DX 59337191 IC50 = 1 nM T65200 C6G1ER 59337195 IC50 = 52 nM T65200 CG5QX1 59337199 IC50 = 7 nM T65200 CXO18I 59337218 IC50 = 2 nM T65200 CW43RZ 59337259 IC50 = 3 nM T65200 C0I9FY 59337265 IC50 = 21 nM T65200 C09NTJ 59337336 IC50 = 357 nM T65200 CLVG32 59337369 IC50 = 30 nM T65200 CM1I5V 59516084 IC50 = 160 nM T65200 C97ATM 59516092 IC50 = 29 nM T65200 CPJ8R9 59635628 IC50 = 0.8 nM T65200 C2ZR8A 59635655 IC50 = 0.8 nM T65200 CLSO80 59635752 IC50 = 5.7 nM T65200 C4BJ0E 59830609 IC50 = 2400 nM T65200 CC05QT 59830625 IC50 = 15 nM T65200 CHL1N8 59830684 IC50 = 520 nM T65200 CDK2F1 59830693 IC50 = 37 nM T65200 C5FX2S 59830700 IC50 = 5 nM T65200 CSHR34 59830789 IC50 = 6 nM T65200 CO60KE 60165516 IC50 = 16 nM T65200 CZPN48 60165517 IC50 = 860 nM T65200 CKB15C 60165655 IC50 = 430 nM T65200 CUSW96 60165656 IC50 = 7 nM T65200 CDY48T 60165657 IC50 = 12 nM T65200 CN6SE1 60165658 IC50 = 170 nM T65200 C1QGN9 60165659 IC50 > 30000 nM T65200 C7XO1R 60165806 IC50 = 120 nM T65200 C4SND8 60167981 IC50 = 1.4 nM T65200 C6GJK8 60167982 IC50 = 1.8 nM T65200 C60PCR 60626745 IC50 = 138 nM T65200 C0ZA5S 66856519 IC50 = 244 nM T65200 C07SOB 67087090 IC50 = 27 nM T65200 C7ID2K 67087238 IC50 = 34 nM T65200 CF1QA5 67087376 IC50 = 12 nM T65200 C93FPL 67463054 IC50 = 3.8 nM T65200 C3G6IP 67464059 IC50 = 18 nM T65200 CG1Y8Z 67464068 IC50 = 4.1 nM T65200 CBT04N 67464726 IC50 = 8.7 nM T65200 C50RPI 67464734 IC50 = 1.8 nM T65200 CVQ7R2 67465177 IC50 = 9.5 nM T65200 C48YEC 67465187 IC50 = 4.1 nM T65200 C1YOA9 67465189 IC50 = 0.9 nM T65200 C6BDM5 67465192 IC50 = 6.8 nM T65200 CG5M4B 67466224 IC50 = 6.6 nM T65200 CNF90O 67466571 IC50 = 3.7 nM T65200 CB73ZN 67466599 IC50 = 3.5 nM T65200 CY83RV 67466819 IC50 = 3.8 nM T65200 C0GEZ6 67467060 IC50 = 58 nM T65200 CY5LT7 67467777 IC50 = 5.4 nM T65200 CU2H4X 67467847 IC50 = 4.6 nM T65200 CXGN47 67467873 IC50 = 6.6 nM T65200 CB05CV 67467924 IC50 = 8.2 nM T65200 CVA0N4 67467988 IC50 = 7.2 nM T65200 CS4ZC0 67468176 IC50 = 27 nM T65200 CJL0P9 67468231 IC50 = 2.2 nM T65200 C2OLT7 67468232 IC50 = 3.7 nM T65200 CJ62MT 67468633 IC50 = 6.8 nM T65200 C8EFA3 67468928 IC50 = 11 nM T65200 CWMX59 68495607 IC50 = 25 nM T65200 C0J7HO 68791928 IC50 = 479 nM T65200 CH4J7L 69021044 IC50 > 22000 nM T65200 C9TPW8 69490242 IC50 = 6.6 nM T65200 C9Z6WC 69491379 IC50 = 106 nM T65200 C0FD9B 69491753 IC50 = 113 nM T65200 CF5J2V 70650743 IC50 = 89 nM T65200 C36OTR 70650937 IC50 = 390 nM T65200 CFA18I 70650942 IC50 = 53 nM T65200 CNPT04 70674215 IC50 = 20 nM T65200 CRS10G 70674564 IC50 = 1 nM T65200 CK0MN8 70674565 IC50 = 1 nM T65200 C3Y6JR 70674566 IC50 = 187 nM T65200 C6Y8BG 70675028 IC50 = 12 nM T65200 CD32VL 70675029 IC50 = 363 nM T65200 CY1Q4D 70675030 IC50 = 360 nM T65200 CC46PN 70675144 IC50 = 1660 nM T65200 CC63NT 70675147 IC50 = 1 nM T65200 CIQC43 70675400 IC50 = 14 nM T65200 CX3Q7I 70681309 IC50 = 22 nM T65200 CJ37ZD 70681407 EC50 = 60 nM T65200 C5XRF0 70681694 IC50 = 21 nM T65200 C35VUM 70681752 IC50 = 1 nM T65200 C5R6QT 70682535 IC50 = 530 nM T65200 COSN63 70682536 IC50 = 7 nM T65200 CV4RM0 70682539 IC50 = 12 nM T65200 CN5KY1 70683408 IC50 = 11 nM T65200 C0SNU2 70683409 IC50 = 1.6 nM T65200 CX4NU3 70683510 EC50 = 802 nM T65200 CLD35R 70683511 EC50 = 3 nM T65200 CAV35N 70683512 EC50 = 1 nM T65200 C3GE8I 70683513 EC50 = 283 nM T65200 CCO71B 70683818 IC50 = 5.3 nM T65200 CQR95L 70683819 IC50 = 3.1 nM T65200 C48WAP 70683820 IC50 = 20 nM T65200 C1Z8FV 70683860 IC50 = 5 nM T65200 CVHB87 70683861 IC50 = 5 nM T65200 COMH43 70683862 IC50 = 351000 nM T65200 CN2Q7K 70684615 IC50 = 430 nM T65200 CNY39A 70684616 IC50 = 17 nM T65200 CJ0EX6 70684625 IC50 = 19 nM T65200 CZ2OC6 70684626 IC50 = 439 nM T65200 C41MYF 70684627 IC50 = 43 nM T65200 C9RJ5T 70685506 IC50 = 3.3 nM T65200 C4FY6J 70685617 EC50 = 55 nM T65200 CNK2P6 70686770 IC50 = 800 nM T65200 CM80QX 70687773 EC50 = 121 nM T65200 CB39WE 70688083 IC50 = 19 nM T65200 C0I5CA 70688084 IC50 = 133 nM T65200 C6B0GN 70688125 IC50 = 14 nM T65200 CLY6C3 70688131 IC50 = 3370 nM T65200 C6GCO3 70688132 IC50 = 50 nM T65200 C7OE6T 70690111 IC50 > 1000 nM T65200 CB1Z6S 70690112 IC50 = 15 nM T65200 CX8I0C 70690113 IC50 = 256 nM T65200 CWF4Q7 70690114 IC50 = 19 nM T65200 CLJ63Y 70690115 IC50 = 61 nM T65200 CB8T1W 70690116 IC50 = 19 nM T65200 C2GUY1 70690164 IC50 = 17 nM T65200 CZI43B 70691963 EC50 = 21 nM T65200 CQ5GB9 70691964 EC50 = 158 nM T65200 C0Q6HK 70692269 IC50 = 652 nM T65200 C6JHM4 70692270 IC50 = 19.1 nM T65200 CLX4T9 70692271 IC50 = 89 nM T65200 C7P6XL 70693999 EC50 = 443 nM T65200 CR2D6E 70694000 EC50 = 4 nM T65200 C7B0TO 70694339 IC50 = 39 nM T65200 CW2UL0 70694375 IC50 = 1 nM T65200 CN1UC6 70695125 IC50 = 100 nM T65200 CJ3QZ7 70695128 IC50 = 5 nM T65200 C2KEZ5 70696021 IC50 = 5.5 nM T65200 CZ9CE1 70696123 EC50 = 686 nM T65200 C56LJT 70696124 EC50 = 90 nM T65200 CI19PU 70696125 EC50 = 47 nM T65200 CX65OK 70696126 EC50 = 70 nM T65200 C0R8AQ 70696127 EC50 = 4 nM T65200 C3M9DS 70696418 IC50 = 27.8 nM T65200 C6RTX3 70696419 IC50 = 33 nM T65200 C9R1UX 70696420 IC50 = 13 nM T65200 CO9B0A 70696421 IC50 = 620 nM T65200 CAIY34 70697161 IC50 = 780 nM T65200 C58PKW 70697162 IC50 = 1300 nM T65200 CWB0C2 70862278 IC50 = 305 nM T65200 CE4HD9 70955517 EC50 = 423 nM T65200 CD5FY6 71249017 IC50 = 10 nM T65200 C8ZKO9 71249030 IC50 = 2 nM T65200 C2JUH6 71449567 IC50 = 3 nM T65200 CESP03 71449568 IC50 = 2 nM T65200 CTW7S1 71449569 IC50 = 14 nM T65200 CL6BC1 71449606 IC50 = 280 nM T65200 C2EL1H 71449988 IC50 = 18 nM T65200 C4XEK5 71449989 IC50 = 260 nM T65200 CS4I5L 71451232 IC50 = 8.4 nM T65200 C64XMB 71451233 IC50 = 11 nM T65200 CTH05X 71451376 IC50 = 107 nM T65200 C03BAV 71451421 IC50 = 385 nM T65200 C6SWH4 71453048 IC50 = 0.4 nM T65200 CCW23U 71453050 IC50 = 17 nM T65200 C2XI0S 71453633 IC50 = 6 nM T65200 CCM5L3 71453634 IC50 = 5 nM T65200 CG13KH 71454792 IC50 = 1800 nM T65200 CJ8Y3Q 71454793 IC50 = 3.1 nM T65200 CIL01G 71454794 IC50 = 9.5 nM T65200 CI2KY5 71454795 IC50 = 6 nM T65200 C74EQT 71454796 IC50 = 43 nM T65200 CJ5EL0 71454844 IC50 = 350 nM T65200 CAM5K2 71454920 IC50 = 4 nM T65200 C6H9GP 71455596 IC50 = 2300 nM T65200 C04FMC 71456569 IC50 = 8400 nM T65200 CZ12EM 71456570 IC50 = 77 nM T65200 C3A2NC 71456571 IC50 = 6.4 nM T65200 C3CAB4 71456572 IC50 = 0.1 nM T65200 C7CVL1 71456573 IC50 = 16 nM T65200 C13AQX 71456704 IC50 = 7 nM T65200 C5AF8Y 71456705 IC50 = 21 nM T65200 CU24OM 71458421 IC50 = 7.7 nM T65200 C9RP6K 71458422 IC50 = 124 nM T65200 CNAM65 71460265 IC50 = 1.5 nM T65200 CLI9G8 71460266 IC50 = 26 nM T65200 CL87SN 71460267 IC50 = 4300 nM T65200 CP5NS2 71460268 IC50 = 3.3 nM T65200 CJ64DO 71460269 IC50 = 5.5 nM T65200 CLGT50 71460270 IC50 = 12 nM T65200 CCBJ60 71460482 IC50 = 118 nM T65200 C8TQF6 71461971 IC50 = 7.2 nM T65200 CYL0P3 71461972 IC50 = 8.2 nM T65200 C94RBY 71461973 IC50 = 3.9 nM T65200 C7HVM9 71462124 IC50 = 1550 nM T65200 C3W7KS 71493483 IC50 = 127 nM T65200 CH1QC0 71493642 IC50 > 300 nM T65200 CCU5S9 71493783 IC50 = 111 nM T65200 CM0I4P 71493785 IC50 = 54.4 nM T65200 CX2Z9F 71493786 IC50 = 73.9 nM T65200 CB7W5K 71493787 IC50 = 83.1 nM T65200 C7FZ5A 71493788 IC50 = 11.9 nM T65200 COTL40 71493931 IC50 = 8.9 nM T65200 C1Q7GU 71493932 IC50 = 25.3 nM T65200 CPO8U3 71493933 IC50 = 3.5 nM T65200 CYD7U3 71493935 IC50 = 36.1 nM T65200 C9SX3J 71493936 IC50 = 10.3 nM T65200 CJ8F6V 71494096 IC50 < 10 nM T65200 C30USY 71511175 IC50 = 0.4 nM T65200 CGE48N 71511231 IC50 = 1 nM T65200 C0D3IO 71511561 IC50 = 0.6 nM T65200 CEC6I8 71540182 IC50 = 43 nM T65200 CHGU58 71540183 IC50 = 104 nM T65200 C7M9AX 71540305 IC50 = 10 nM T65200 C04NSW 71540306 IC50 = 2 nM T65200 CIE32C 71542765 IC50 = 10.5 nM T65200 CIB90N 71579771 EC50 > 10000 nM T65200 C5V7BA 71579772 EC50 = 21 nM T65200 C1J4BE 71579773 EC50 = 213 nM T65200 CF4UA2 71579774 EC50 = 1980 nM T65200 C1N9YA 71579775 EC50 = 194 nM T65200 CI7XN8 71579776 EC50 = 0.03 nM T65200 CWMP51 71579867 EC50 = 72 nM T65200 CCEJ75 71579868 EC50 = 49 nM T65200 CHQ03A 71579869 EC50 = 604 nM T65200 CRY78W 71652334 IC50 = 92 nM T65200 CF1I4V 71652335 IC50 = 793 nM T65200 CXYU90 71652498 IC50 = 621 nM T65200 CC8V9G 71652499 IC50 > 1000 nM T65200 CA2B9L 71652500 IC50 > 1000 nM T65200 CT34MK 71652501 IC50 = 956 nM T65200 C15HXP 71652502 IC50 = 277 nM T65200 C4U6YN 71652503 IC50 = 825 nM T65200 CX7FW3 71652656 IC50 = 310 nM T65200 CW2P7F 71652657 IC50 > 1000 nM T65200 C3MK2C 71654170 IC50 = 1316 nM T65200 CH19CW 71654171 IC50 = 945 nM T65200 CAN6L8 71654173 IC50 = 594 nM T65200 CDXS16 71654174 IC50 = 107 nM T65200 CK1P2H 71654341 IC50 = 27 nM T65200 CBL81E 71654342 IC50 = 2373 nM T65200 CZ0X8N 71654493 IC50 = 853 nM T65200 CYG2V8 71654494 IC50 = 741 nM T65200 CD5C1E 71654495 IC50 = 277 nM T65200 CU5SX2 71654496 IC50 = 28 nM T65200 C5ST2Z 71654497 IC50 = 3.3 nM T65200 C3K9FA 71654658 IC50 = 659 nM T65200 CP2FO3 71654659 IC50 = 715 nM T65200 C0G3PT 71654661 IC50 = 141 nM T65200 C3GYJ9 71654663 IC50 = 1484 nM T65200 C6WYZ2 71654664 IC50 = 71 nM T65200 CS62EO 71716496 IC50 = 11.1 nM T65200 CKE1O8 71716497 IC50 = 19.8 nM T65200 CWEU78 71717721 IC50 = 6.7 nM T65200 CGQ3N4 71718328 IC50 = 13 nM T65200 CC1S7O 71718329 IC50 = 9.8 nM T65200 C17HUV 71718928 IC50 = 11.1 nM T65200 CG07AZ 71718929 IC50 = 8 nM T65200 CLP4Q7 71719544 IC50 = 3.8 nM T65200 CK7I1V 71719545 IC50 < 3 nM T65200 CLS72I 71720140 IC50 = 29.3 nM T65200 CC07BN 71720785 IC50 = 5.4 nM T65200 CTAQ96 71720786 IC50 = 39.3 nM T65200 CPW3L4 71745145 IC50 = 11400 nM T65200 C0RE2C 71745149 IC50 = 3200 nM T65200 CZO20P 71813157 IC50 = 675 nM T65200 CZ1AD6 72188908 IC50 = 27200 nM T65200 C2Q6YJ 72670421 IC50 = 4 nM T65200 CV51GE 72792443 IC50 = 3.7 nM T65200 C0WCX4 72793118 IC50 > 1000000 nM T65200 CBC58T 73112834 IC50 = 89 nM T65200 C1AS0K 73212955 IC50 = 1929 nM T65200 CV4CT7 73213039 IC50 = 85 nM T65200 C16EOU 73213122 IC50 = 449 nM T65200 CH1JK9 73213123 IC50 = 4.8 nM T65200 C4ZEJ5 73213208 IC50 = 4080 nM T65200 CHC25V 73213209 IC50 = 282 nM T65200 CLMD08 73213210 IC50 = 107 nM T65200 C1ODB9 73213211 IC50 = 640 nM T65200 CCFW14 73213282 IC50 = 26 nM T65200 C0GC9K 73213283 IC50 = 190 nM T65200 C1Z3RN 73213342 IC50 = 6 nM T65200 C8Y0SL 73213343 IC50 = 2 nM T65200 C8ZH3R 73213344 IC50 = 2.6 nM T65200 CIL79J 73213345 IC50 = 2.3 nM T65200 CJAH38 73213346 IC50 = 8 nM T65200 C2WSB1 73213403 IC50 = 8 nM T65200 CR4NF8 73213404 IC50 = 20 nM T65200 CFH37L 73213405 IC50 = 5 nM T65200 CT3WK7 73213406 IC50 = 14 nM T65200 CXKG30 73213407 IC50 = 102 nM T65200 CYAJ36 73345978 IC50 = 266.1 nM T65200 CO7R8B 73347331 IC50 = 9 nM T65200 CAV13P 73348835 IC50 = 11 nM T65200 CZ1V0X 73350418 IC50 = 14 nM T65200 CIO4G6 73350419 IC50 = 9 nM T65200 CG15WM 73352110 IC50 = 330.8 nM T65200 CALM65 73352112 IC50 = 165.4 nM T65200 C46KTL 73353391 IC50 = 4 nM T65200 C9WA7F 73353568 IC50 = 249 nM T65200 CJ3O7S 73353624 IC50 = 31 nM T65200 CV72YC 73355069 IC50 = 407.3 nM T65200 CGR3P5 73355072 IC50 = 116.4 nM T65200 C3DJ5W 73356463 IC50 = 18 nM T65200 C32YFH 73356464 IC50 = 19 nM T65200 C6HBS9 73356465 IC50 = 9 nM T65200 C15SEC 73356624 IC50 = 9.4 nM T65200 C2FOM5 73356626 IC50 = 403700 nM T65200 CV70BR 73356628 IC50 = 910 nM T65200 CWC4Z5 73356629 IC50 = 770.6 nM T65200 C34DYM 74369475 IC50 = 64 nM T65200 C0ATV1 74369476 IC50 = 32 nM T65200 C96KTM 76311127 IC50 = 1.5 nM T65200 C7SL8F 76311128 IC50 = 69 nM T65200 CM7Z1F 76311129 IC50 = 50 nM T65200 CLSC64 76311130 IC50 = 153 nM T65200 C8B7QC 76314399 IC50 = 57 nM T65200 CD59ZS 76314744 IC50 = 4.4 nM T65200 CHC37L 76314745 IC50 = 1.3 nM T65200 C3W6KR 76314746 IC50 = 12 nM T65200 C2A1EZ 76318320 IC50 = 9.9 nM T65200 CFIG02 76318321 IC50 = 2.8 nM T65200 C2MN9P 76318322 IC50 = 0.43 nM T65200 CH2Z3V 76318323 IC50 = 2090 nM T65200 CGW47O 76318324 IC50 = 216 nM T65200 CWM24C 76318325 IC50 = 8600 nM T65200 CRD2G3 76321050 IC50 = 8 nM T65200 CJ7IB1 76322005 IC50 = 0.4 nM T65200 C0S2AR 76322006 IC50 = 0.49 nM T65200 C5LVE9 76322007 IC50 = 13 nM T65200 CAP0Q9 76322008 IC50 = 9 nM T65200 C57VPS 76322009 IC50 = 8.1 nM T65200 C4L0JB 76322010 IC50 = 14 nM T65200 CTJQ98 76322011 IC50 = 3.6 nM T65200 CK8WD4 76322012 IC50 = 48 nM T65200 CRD0H3 76322013 IC50 > 20500 nM T65200 C7RA5E 76322014 IC50 = 29 nM T65200 C3FHA2 76322015 IC50 = 104 nM T65200 CJV62C 76325306 IC50 = 1 nM T65200 CN8MZ5 76325631 IC50 = 1.7 nM T65200 CFGC62 76325632 IC50 = 43 nM T65200 CS4Z6D 76325633 IC50 = 47 nM T65200 C63SQI 76328857 IC50 = 2 nM T65200 C4PHX5 76329207 IC50 = 486 nM T65200 CD63UM 76329208 IC50 = 18 nM T65200 CH0A4M 76329209 IC50 = 10 nM T65200 CBM38K 76329210 IC50 = 230 nM T65200 CM8BP5 76331939 IC50 = 2 nM T65200 C48NWX 76332527 IC50 = 7 nM T65200 C5F7PO 76332860 IC50 = 1.7 nM T65200 C1OD3M 76332861 IC50 = 45 nM T65200 C1AU3Y 76332862 IC50 = 142 nM T65200 CS1MD9 76336472 IC50 = 0.4 nM T65200 C1U4LO 76336473 IC50 = 28 nM T65200 CWBL78 76336474 IC50 = 23 nM T65200 CO90PM 76336475 IC50 = 13 nM T65200 C4Q3GC 76336476 IC50 = 10 nM T65200 CD3S8Z 90294149 IC50 = 0.2 nM T65200 C01ICD 90294162 IC50 > 1000 nM T65200 C0L5YD 90643786 IC50 = 1 nM T65200 CPN65E 90643787 IC50 = 4 nM T65200 C8MY4O 90643788 IC50 = 3200 nM T65200 CSHC95 90643789 IC50 = 1.2 nM T65200 CB5Z1O 90643790 IC50 = 0.4 nM T65200 C9DCJ5 90643791 IC50 = 6 nM T65200 CPIJ68 90643792 IC50 = 74 nM T65200 CRH23E 90643793 IC50 = 100 nM T65200 CZ6L4V 90644192 IC50 = 15 nM T65200 COWH43 90666511 IC50 = 326 nM T65200 CH2V5Y 90666512 IC50 = 576 nM T65200 C2K5HD 90666513 IC50 = 290 nM T65200 C8IV9K 90666515 IC50 = 215 nM T65200 CS1L3X 90666516 IC50 = 582 nM T65200 C6JF9M 90666517 IC50 = 332 nM T65200 C9XP2Z 90666525 IC50 = 401 nM T65200 CEU5D8 90667160 IC50 = 26 nM T65200 CGFN76 90667161 IC50 = 10 nM T65200 CPAB18 90667162 IC50 = 7 nM T65200 CQ7YM9 90667163 IC50 = 6 nM T65200 CQ0K6M 90667192 IC50 = 910 nM T65200 CPB5Y9 90667193 IC50 > 30000 nM T65200 C58GBO 90667194 IC50 = 280 nM T65200 CNFW97 90667195 IC50 = 91 nM T65200 CK1Z9Y 90667196 IC50 = 200 nM T65200 C1XHM9 90667197 IC50 = 300 nM T65200 CRK73P 90667198 IC50 = 150 nM T65200 C9Z1JM 90667199 IC50 = 110 nM T65200 CZW6V9 90667200 IC50 = 29 nM T65200 CR6QE2 90667201 IC50 = 57 nM T65200 CS34ET 90667202 IC50 = 13000 nM T65200 CJ9L0F 90667203 IC50 = 76 nM T65200 C8XFR7 90667204 IC50 = 660 nM T65200 C0P7FQ 90667205 IC50 = 400 nM T65200 CGM3N0 90667206 IC50 = 57 nM T65200 CRM06S 90667207 IC50 = 6000 nM T65200 C0C5LA 90667208 IC50 = 280 nM T65200 CZ0V7B 90667209 IC50 = 86 nM T65200 CJ30KP 90667210 IC50 = 180 nM T65200 CX19FE 90667211 IC50 = 3000 nM T65200 CCW9F0 90667212 IC50 = 110 nM T65200 CD8Y7M 90667213 IC50 = 79 nM T65200 CMG8X0 90667214 IC50 = 33 nM T65200 CQ23WR 90667215 IC50 = 98 nM T65200 CQ6G7I 90667216 IC50 = 6300 nM T65200 CZOY61 90667217 IC50 > 30000 nM T65200 C5GS6J 90667218 IC50 = 2100 nM T65200 C62OKJ 90667219 IC50 > 30000 nM T65200 CM7L9J 90667220 IC50 = 900 nM T65200 C4UO9B 90667221 IC50 > 30000 nM T65200 CN8U0J 90667222 IC50 = 830 nM T65200 CJN9U1 90667223 IC50 = 2800 nM T65200 C59XZL 90667224 IC50 = 200 nM T65200 CM2H3Q 90667225 IC50 = 2500 nM T65200 C9QZE2 91039859 IC50 = 0.61 nM T65200 CFSK10 101911911 IC50 = 194.5 nM T65200 CO0H9S 101911912 IC50 = 15.3 nM T65200 C91CLR 101911913 IC50 = 75.5 nM T65200 C9RBA1 101911914 IC50 = 395.2 nM T65200 CMOG09 101911915 IC50 = 34.1 nM T65200 C2EL1D 101914701 IC50 = 10000 nM T65200 C50GBO 102528497 IC50 > 1000000 nM T65200 CR0F4L 108452142 IC50 = 50 nM T65200 C6JK4C 118034965 IC50 = 25 nM T65200 C54FXC 118034981 IC50 = 6 nM T65200 CV37ZA 118035109 IC50 = 2 nM T65200 C6QV4O 118035249 IC50 > 1000 nM T65200 C1SHM4 118035255 IC50 > 1000 nM T65200 CE4C3S 118035314 IC50 > 1000 nM T65200 CYS71J 118035319 IC50 = 15 nM T65200 C0EJ2D 118035332 IC50 > 1000 nM T65200 CEB27J 118035356 IC50 > 1000 nM T65200 C7XTF5 118035368 IC50 = 34 nM T65200 CD1RX4 118035384 IC50 = 0.3 nM T65200 CX19FR 118035469 IC50 = 9 nM T65200 C2WPZ9 118707674 IC50 = 8100 nM T65200 CU7BI0 118707675 IC50 = 13000 nM T65200 CL8QZ9 118709251 IC50 = 1.7 nM T65200 C3AE6V 118709252 IC50 = 8.1 nM T65200 C1T2CF 118709253 IC50 = 20 nM T65200 CDQV28 118709254 IC50 = 42 nM T65200 CV21FA 118709255 IC50 = 65 nM T65200 C9S7KJ 118709256 IC50 = 51 nM T65200 CGS20Q 118709257 IC50 = 4.2 nM T65200 C1N3VB 118709258 IC50 = 2.4 nM T65200 CMX6S5 118709259 IC50 = 13 nM T65200 CC79WV 118709260 IC50 = 17 nM T65200 CY6HN5 118713835 IC50 = 10000 nM T65200 C5NP3O 118713838 IC50 = 10000 nM T65200 C8WIS4 118713840 IC50 = 10000 nM T65200 CGNW12 118715853 IC50 = 79 nM T65200 CO9TR1 118715854 IC50 = 21000 nM T65200 CH1QF3 118723425 IC50 = 1400 nM T65200 CJN94G 118723426 IC50 = 4100 nM T65200 CS41LP 118723427 IC50 = 3800 nM T65200 CLN78Y 118723428 IC50 = 2300 nM T65200 CL8TD4 118728612 IC50 = 5.3 nM T65200 CZF5Y1 122186854 IC50 = 14 nM T65200 CI3QS6 122186855 IC50 > 1000 nM T65200 C2GU9V 122186856 IC50 = 55 nM T65200 CP3JF2 122187896 IC50 = 28 nM T65200 CM3E5Z 122187897 IC50 > 1000 nM T65200 C73BLA 122187898 IC50 > 1000 nM T65200 C60BFG 122187899 IC50 > 1000 nM T65200 C9FZ3G 122187900 IC50 > 1000 nM T65200 CM2SE3 122187901 IC50 = 2 nM T65200 CHG3Q6 122187902 IC50 = 44 nM T65200 CH5Q2J 122187903 IC50 > 1000 nM T65200 CFU94A 122187904 IC50 = 0.1 nM T65200 CWRU87 122189728 IC50 = 74 nM T65200 C6FVO4 127026799 IC50 > 1000000 nM T65200 CS7H8G 127026800 IC50 > 1000000 nM T65200 C95CJO 127026801 IC50 > 1000000 nM T65200 CKWX64 127027103 IC50 > 1000000 nM T65200 CVK76L 127027104 IC50 > 1000000 nM T65200 CO19WK 127027115 IC50 > 1000000 nM T65200 CQ9UV5 127027406 IC50 > 1000000 nM T65200 C3CLW7 127027407 IC50 > 1000000 nM T65200 C86HRL 127027408 IC50 > 1000000 nM T65200 C5K2HO 127027409 IC50 > 1000000 nM T65200 C7RD3B 127037645 IC50 = 100 nM T65200 CF3DC8 127037646 IC50 = 1000 nM T65200 C4YZD2 127037647 IC50 = 19.95 nM T65200 CZA2B7 127037648 IC50 = 63.1 nM T65200 C8VNT6 127037649 IC50 = 31.62 nM T65200 CISV60 127037668 IC50 = 31.62 nM T65200 CV2UK8 127037669 IC50 = 251.19 nM T65200 COW9D0 127037670 IC50 = 316.23 nM T65200 CC49JY 127037671 IC50 = 501.19 nM T65200 C0QH3O 127037762 IC50 = 1078 nM T65200 C0D9OG 127037764 IC50 = 267 nM T65200 C51EXJ 127037765 IC50 = 12180 nM T65200 C7WYI8 127037831 IC50 = 94000 nM T65200 CO0J6N 127037847 IC50 > 1000000 nM T65200 CI5HA6 127037875 IC50 > 1000000 nM T65200 C1T6JY 127037989 IC50 = 50.12 nM T65200 CAE17F 127037991 IC50 = 3853 nM T65200 C15LKR 127038025 IC50 = 19.95 nM T65200 CP0JV9 127038197 IC50 = 245000 nM T65200 CRQZ81 127038201 IC50 > 1000000 nM T65200 CWF34T 127038235 IC50 > 1000000 nM T65200 CA8Q4V 127038358 IC50 = 63.1 nM T65200 C0Z4RN 127038441 IC50 = 60 nM T65200 C7VA1T 127038442 IC50 = 459 nM T65200 C2B8WY 127038443 IC50 = 1515 nM T65200 C5GKD3 127038444 IC50 = 201 nM T65200 C5VDS8 127038445 IC50 = 2659 nM T65200 CN5ZC3 127038533 IC50 > 1000000 nM T65200 CS7KZ0 127038549 IC50 > 1000000 nM T65200 CZI59Q 127038555 IC50 > 1000000 nM T65200 COQ0Y7 127038824 IC50 = 15 nM T65200 C8K2LF 127038877 IC50 > 1000000 nM T65200 CB7DA8 127039136 IC50 = 26 nM T65200 C6BH8N 127039137 IC50 = 32 nM T65200 CYHP24 127039138 IC50 = 22 nM T65200 CUBG78 127039139 IC50 = 8 nM T65200 C2YRT8 127039140 IC50 = 40 nM T65200 CPT7I8 127039141 IC50 = 40 nM T65200 CV71AT 127039204 IC50 > 1000000 nM T65200 C1PMH2 127039211 IC50 > 1000000 nM T65200 C4MLS1 127039230 IC50 > 1000000 nM T65200 C0Y9XU 127039453 IC50 = 89 nM T65200 CDT2U8 127039457 IC50 = 12 nM T65200 C28IXT 127039458 IC50 = 57 nM T65200 CFA46N 127039459 IC50 = 25 nM T65200 CO9K6F 127039460 IC50 = 11 nM T65200 C0L8QG 127039859 IC50 > 1000000 nM T65200 CB5E9Z 127040446 IC50 = 63.1 nM T65200 CTK29W 127040447 IC50 = 50.12 nM T65200 C0FIK4 127040448 IC50 = 25.12 nM T65200 CO6FR3 127040449 IC50 = 10 nM T65200 CR2AB4 127040450 IC50 = 15.85 nM T65200 CB67GJ 127040451 IC50 = 63.1 nM T65200 C4E1LF 127040565 IC50 > 1000000 nM T65200 CTN4E7 127040566 IC50 > 1000000 nM T65200 CLB1N5 127040732 IC50 = 648 nM T65200 C6MY2R 127040750 IC50 = 6.31 nM T65200 C4JQ2N 127040751 IC50 = 25.12 nM T65200 C4KPO7 127040752 IC50 = 25.12 nM T65200 CK43ZL 127040753 IC50 = 50.12 nM T65200 C3MH6O 127040764 IC50 = 398.11 nM T65200 CB67LT 127040901 IC50 = 341000 nM T65200 C5P3KE 127040902 IC50 > 1000000 nM T65200 CT5Q1A 127040903 IC50 > 1000000 nM T65200 CW3FN4 127040904 IC50 > 1000000 nM T65200 C9EQX2 127040905 IC50 = 33000 nM T65200 C32ADQ 127040906 IC50 > 1000000 nM T65200 CDFO34 127040907 IC50 > 1000000 nM T65200 CO1RS3 127041085 IC50 = 199.53 nM T65200 CVRU05 127041086 IC50 = 10 nM T65200 CWD5G7 127041087 IC50 = 15.85 nM T65200 C8ED4P 127041144 IC50 = 1000 nM T65200 C42PNF 127041145 IC50 = 350 nM T65200 C4O8QH 127041220 IC50 > 1000000 nM T65200 CC7QS3 127041221 IC50 > 1000000 nM T65200 C4BGE0 127041222 IC50 > 1000000 nM T65200 CVP7A1 127041223 IC50 > 1000000 nM T65200 CG9Q2T 127041801 IC50 > 1000000 nM T65200 CYNI06 127041808 IC50 > 1000000 nM T65200 C1ZUD5 127041809 IC50 > 1000000 nM T65200 CCU4H6 127041810 IC50 = 122000 nM T65200 CZN2A0 127041811 IC50 = 8000 nM T65200 CFR23K 127041837 IC50 > 1000000 nM T65200 C0ZC4E 127041838 IC50 > 1000000 nM T65200 CGOB70 127041839 IC50 > 1000000 nM T65200 CCKL17 127042099 IC50 = 74000 nM T65200 C24EQS 127042100 IC50 = 121000 nM T65200 CE64CI 127042101 IC50 > 1000000 nM T65200 COR6A5 127042102 IC50 > 1000000 nM T65200 C7Y4XU 127042440 IC50 > 1000000 nM T65200 CKM3I9 127042477 IC50 > 1000000 nM T65200 CMP75K 127042478 IC50 > 1000000 nM T65200 C0WXN2 127042636 IC50 > 1000000 nM T65200 C41CMW 127042637 IC50 > 1000000 nM T65200 CD1VZ3 127042638 IC50 > 1000000 nM T65200 CMCP64 127042780 IC50 = 18000 nM T65200 C4OUL9 127042781 IC50 = 85000 nM T65200 C7XI3U 127042782 IC50 > 1000000 nM T65200 CRE59A 127042783 IC50 > 1000000 nM T65200 CRP78U 127042784 IC50 > 1000000 nM T65200 C6AHS2 127042785 IC50 > 1000000 nM T65200 C1LMV6 127042786 IC50 > 1000000 nM T65200 C0CG7T 129245779 IC50 = 197 nM T65200 C2S1IG 129245927 IC50 = 496 nM T65200 C52OSA 129246019 IC50 = 902 nM T65200 CC7KT2 129246025 IC50 = 373 nM T65200 C0X2PF 129246036 IC50 = 266 nM T65200 C8FRH7 131750120 IC50 = 0.7 nM T65200 CC2G0S 132045061 IC50 = 1490 nM T65200 CGWV92 132053849 IC50 = 30 nM T65200 CT05EL 135399889 Ki = 14 nM T65200 CI4W7U 135411280 IC50 = 1950 nM T65200 CTS3H5 135416151 IC50 = 1102 nM T65200 CXCZ71 135427920 IC50 = 3.9 nM T65200 C02KAD 135440148 IC50 = 2.8 nM T65200 CE0S3Y 135465949 IC50 = 1.8 nM T65200 CU3V4A 135478350 IC50 = 7980 nM T65200 CM7A1J 135492551 IC50 = 2 nM T65200 CN9X3Y 135513260 IC50 = 20 nM T65200 C94SLQ 135513261 Ki = 130 nM T65200 C5D7BR 135513262 IC50 = 40 nM T65200 C6L5UI 135513263 Ki = 18 nM T65200 CB3YH5 135513264 Ki = 7 nM T65200 C8EF7V 135513265 Ki = 4 nM T65200 CS6I2E 135513267 Ki = 48 nM T65200 CBA2F6 135513268 Ki = 22 nM T65200 CV2I5D 135513269 IC50 = 53 nM T65200 CUC4R9 135513270 Ki = 87 nM T65200 CAI18X 135513271 Ki = 8 nM T65200 C1YW0Z 135513272 Ki = 9 nM T65200 CJ7Z5X 135513273 IC50 = 18 nM T65200 CKES51 135556845 Ki = 30 nM T65200 CYN12P 135559069 Ki = 3 nM T65200 C0NY3F 135559070 Ki = 20 nM T65200 CLW3Y7 135566336 Ki = 7 nM T65200 CBQM57 135566449 IC50 = 34 nM T65200 CQ7K2C 135566823 IC50 = 24 nM T65200 C2AG1T 135567651 IC50 = 2250 nM T65200 CE2JP5 135588530 IC50 = 1090 nM T65200 C9A7BT 135590905 Ki = 220 nM T65200 C7H1IV 135590907 Ki = 26 nM T65200 C9VH4K 135610998 Ki = 120 nM T65200 CNW10S 135611019 Ki = 76 nM T65200 C1UR6Y 135611029 Ki = 1800 nM T65200 C98OIC 135611051 IC50 = 32 nM T65200 CCQJ43 135611106 IC50 = 18 nM T65200 C13XPC 135611120 Ki = 44 nM T65200 C2K9OD 135611129 IC50 = 11 nM T65200 CGZT41 135611130 Ki = 28 nM T65200 C4YO9E 135612240 IC50 = 0.34 nM T65200 CB6U1X 135783315 Ki = 126 nM T65200 C04ELB 135783316 Ki = 55 nM T65200 C61NUT 135783317 Ki = 64 nM T65200 CB76YU 135783318 Ki = 34 nM T65200 C76MEG 135783319 Ki = 82 nM T65200 CMQ2L1 135783320 Ki = 32 nM T65200 CE6L4S 135783321 Ki = 47 nM T65200 CTAM34 135783322 Ki = 28 nM T65200 CV6KJ5 135783323 Ki = 58 nM T65200 CG03DH 135783324 Ki = 38 nM T65200 C7B3JV 135783325 Ki = 73 nM T65200 C0PZ2W 135783326 Ki = 25 nM T65200 CUL73D 135783327 Ki = 372 nM T65200 C59KXI 135783328 Ki = 149 nM T65200 CKB54L 135783329 Ki = 13 nM T65200 CB93HT 135783330 Ki = 12 nM T65200 C9SX2F 135783331 Ki = 24 nM T65200 CXE02J 135783332 Ki = 24 nM T65200 C7ZTC5 135783333 Ki = 26 nM T65200 C09UQY 135783334 Ki = 13 nM T65200 CL5F0J 135783335 Ki = 3 nM T65200 CPB81K 135783336 Ki = 20 nM T65200 CTP32F 135783337 Ki = 28 nM T65200 CQ3LU8 135796677 Ki = 20 nM T65200 C3K6QX 135796678 Ki = 369 nM T65200 C3EF0Q 135857018 Ki = 22 nM T65200 C97JHG 135857019 Ki = 3500 nM T65200 CDE06Q 135857020 Ki = 240 nM T65200 CZT73E 135857021 Ki = 330 nM T65200 CN71RY 135857022 Ki = 46 nM T65200 C36WCX 135857023 Ki = 84 nM T65200 CS2KM5 135857025 Ki = 83 nM T65200 CJ4EC8 135857030 Ki = 79 nM T65200 C0X9LJ 135857031 Ki = 60 nM T65200 CSXM30 135857032 Ki = 210 nM T65200 C6I8MT 135857033 IC50 = 78 nM T65200 C2C0QF 135857034 IC50 = 180 nM T65200 CA2ZD0 135857035 Ki = 34 nM T65200 CV64MY 135857036 Ki = 25 nM T65200 CB1S9P 135857038 Ki = 290 nM T65200 CYQV73 135857043 Ki = 210 nM T65200 C1BT9R 135857054 Ki = 6500 nM T65200 CKG8Y7 135857055 Ki = 130 nM T65200 C87VBH 135857056 Ki = 100 nM T65200 CPH26Z 135870734 IC50 = 8.511 nM T65200 CSTE94 135890077 Ki = 329 nM T65200 CFM10Y 135890078 Ki = 227 nM T65200 CL94TI 135890089 IC50 = 12.6 nM T65200 C4UI0T 135890090 Ki = 27.8 nM T65200 C0M2BY 135890091 Ki = 30.6 nM T65200 C5R9GE 135890092 Ki = 47.2 nM T65200 CBTS50 135950092 Ki = 22 nM T65200 CI9O6Z 135950093 Ki > 10000 nM T65200 CQP26U 135950094 Ki = 1433 nM T65200 CC43KF 135950095 Ki = 17 nM T65200 C2HBT1 135950096 Ki = 17 nM T65200 CHOQ23 135950097 Ki = 14 nM T65200 C8UCN0 135950098 Ki = 7 nM T65200 C1UJQ2 135950099 Ki = 12 nM T65200 CJR3T2 135950100 Ki = 6 nM T65200 CSX5A2 135950101 Ki = 18 nM T65200 C32DMH 135950103 Ki = 6 nM T65200 C5POA0 135950104 Ki = 4 nM T65200 CUV4I5 135950105 Ki = 43 nM T65200 CTP6Z0 135950106 Ki = 39 nM T65200 C6U8FG 135950107 Ki = 25 nM T65200 C0ZV4L 135950110 Ki = 879 nM T65200 C82WYA 135967653 IC50 = 120 nM T65200 C7SZW5 135967654 IC50 = 47 nM T65200 C6IYH3 135967877 IC50 = 358 nM T65200 C0FO4G 135980568 IC50 = 504 nM T65200 C1L7CK 135989418 IC50 = 12.7 nM T65200 C4Q2VX 135989508 Ki = 6 nM T65200 CK6QW9 135989522 IC50 = 10.2 nM T65200 CZ3D8G 135989534 IC50 = 15 nM T65200 CX3VU1 136000590 IC50 = 8.8 nM T65200 CNQ25Z 136021384 IC50 = 51 nM T65200 CXQ8H4 136036583 IC50 = 89 nM T65200 C4S0JG 136060656 Ki = 77 nM T65200 CV3K8F 136060657 Ki = 676 nM T65200 CW9A7N 136060658 Ki = 871 nM T65200 CN1J8U 136060659 Ki = 1418 nM T65200 CKE5L0 136060660 Ki > 10000 nM T65200 CHA4P2 136060661 Ki > 10000 nM T65200 C0DYV7 136060662 Ki > 10000 nM T65200 C9S1IO 136060663 Ki = 2875 nM T65200 C1YP4J 136060664 Ki = 19 nM T65200 CY4BX8 136060665 IC50 = 12 nM T65200 CAGT25 136060680 IC50 = 97 nM T65200 C7W4GE 136088954 IC50 = 38 nM T65200 CT3RN8 136141565 IC50 = 140 nM T65200 C03UTQ 136169588 Ki = 151 nM T65200 CDL2N0 136183479 IC50 = 177 nM T65200 CR74OZ 136188845 IC50 > 40000 nM T65200 CMF49E 136219287 IC50 = 215 nM T65200 C7O0AF 136219288 IC50 = 50 nM T65200 C9V3GU 136219289 IC50 = 652 nM T65200 CIWC75 136219290 IC50 = 15 nM T65200 C2G8OB 136219291 IC50 = 197 nM T65200 CB8A3D 136219292 IC50 = 1220 nM T65200 CB01IL 136219293 IC50 = 406 nM T65200 CA54EM 136219294 IC50 = 4 nM T65200 CV73MH 136219295 IC50 = 27 nM T65200 C8QY2P 136239322 IC50 = 28 nM T65200 CSC95T 136239323 IC50 = 18 nM T65200 CUK9O4 136239324 IC50 = 80 nM T65200 C5ZU7W 136239325 IC50 = 63 nM T65200 CF29MI 136239456 IC50 = 6 nM T65200 C74JBX 136239457 IC50 = 10 nM T65200 C45XPI 136239458 IC50 = 234 nM T65200 CSN75O 136239459 IC50 > 2250 nM T65200 C43VJL 136239460 IC50 = 64 nM T65200 C69KXC 136244467 IC50 = 1480 nM T65200 C09OKY 136244468 IC50 = 11 nM T65200 COE1D8 136244469 IC50 = 7 nM T65200 C5O9YE 136244470 IC50 = 7 nM T65200 C73KLZ 136244471 IC50 = 22 nM T65200 CQUE75 136244472 IC50 = 13 nM T65200 CU72CG 136244473 IC50 = 11 nM T65200 C7RW8H 136244474 IC50 = 65 nM T65200 CQ2F0N 136244563 IC50 = 4 nM T65200 C0RE7P 136244564 IC50 = 575 nM T65200 C6EUA9 136244565 IC50 = 425 nM T65200 C1VF3O 136244566 IC50 = 671 nM T65200 C3SI8Z 136254198 IC50 = 237 nM T65200 C23BLV 136254199 Ki = 37.3 nM T65200 CU0H5S 136254200 Ki = 27 nM T65200 C9M3JP 136254201 Ki = 17.5 nM T65200 CHWB52 136254421 IC50 = 4 nM T65200 C57EKM 136254422 IC50 = 38 nM T65200 CY8KQ9 136254423 IC50 = 1580 nM T65200 CXEP17 136254424 IC50 = 334 nM T65200 CBZ43H 136254425 IC50 = 82 nM T65200 CA08JL 136254426 IC50 > 2250 nM T65200 CK4ZV2 136254427 IC50 > 2250 nM T65200 CM07SD 136254428 IC50 = 24 nM T65200 CH7ED9 136260445 IC50 > 2250 nM T65200 CYM96W 136260446 IC50 = 139 nM T65200 CS73EM 136260447 IC50 = 655 nM T65200 C48VPD 136260448 IC50 = 799 nM T65200 CSIF40 136260449 IC50 = 16 nM T65200 C51JWX 136260516 IC50 = 18 nM T65200 C8I9XD 136260517 IC50 = 4 nM T65200 CD9BM2 136260518 IC50 = 104 nM T65200 CM8Z3R 136260519 IC50 = 8 nM T65200 CSQC20 137632531 IC50 = 40 nM T65200 CZ1IK0 137637149 IC50 = 531 nM T65200 CC70AR 137637699 IC50 = 14 nM T65200 CWJ0X4 137637923 IC50 = 729 nM T65200 CB1LR0 137638399 IC50 = 101 nM T65200 CKO2B8 137641803 IC50 = 488 nM T65200 CGC8D6 137642286 IC50 = 66 nM T65200 C7W6ST 137642412 IC50 = 919 nM T65200 CQJA02 137644192 IC50 = 244 nM T65200 C1D8PB 137647393 IC50 = 13 nM T65200 CBV52L 137649348 IC50 = 148 nM T65200 CZ59OU 137650452 IC50 = 4 nM T65200 CDS86M 137656441 IC50 = 1047 nM T65200 C94RSY 137656587 IC50 = 994 nM T65200 CD94IC 137659160 IC50 = 1 nM T65200 C0DHM9 145952000 IC50 = 20 nM T65200 C2M3UR 145952031 IC50 = 290 nM T65200 CC91LF 145952333 IC50 = 90 nM T65200 CY59DH 145953557 IC50 = 410 nM T65200 CWA0O3 145953890 IC50 = 40 nM T65200 C0YZ9H 145955053 IC50 = 2770 nM T65200 CDT3Q6 145956314 IC50 = 20 nM T65200 C97ENK 145957179 IC50 = 1220 nM T65200 C09QUS 145958039 IC50 = 20 nM T65200 CZ1I4O 145958159 IC50 = 320 nM T65200 C8MDL6 145960048 IC50 = 1080 nM T65200 CV6Q5J 145960157 IC50 = 30 nM T65200 C9IQK7 145980859 IC50 = 1620 nM T65200 CMVS94 155512106 Ki = 270 nM T65200 C1F9PV 155515115 Ki = 353700 nM T65200 CPO9M4 155520336 Ki = 145000 nM T65200 CXOU89 155521135 Ki = 4630 nM T65200 C8WNT0 155521284 Ki = 210 nM T65200 CN59WH 155525513 Ki = 289000 nM T65200 C1D4WM 155537728 Ki = 11800 nM T65200 CV5KQ0 155543491 Ki = 5000 nM T65200 CKFU03 155545095 Ki = 130000 nM T65200 CG19XT 155548236 Ki = 5150 nM T65200 CB08IM 155548826 Ki = 13500 nM T65200 C1GC0O 155553184 Ki = 24000 nM T65200 C4MHK6 155555049 IC50 = 1900 nM T65200 CEM03Y 155556588 Ki = 8230 nM T65200 C9E6AM 155561480 Ki = 57600 nM T65200 COWH25 155562798 IC50 > 500000 nM T65200 CM3TZ5 155563780 IC50 = 9900 nM T65200 CZT7P4 155567250 Ki = 21200 nM T65200 D00DDJ 17233943 IC50 = 8200 nM T65200 D00PSW 3630776 IC50 = 7.5 nM T65200 D00QOL 11673314 IC50 = 107 nM T65200 D01CAC 45269321 IC50 = 111 nM T65200 D01EBV 21672621 IC50 = 5200 nM T65200 D02KXX 586971 IC50 = 200 nM T65200 D02WUU 15627039 IC50 = 102 nM T65200 D03JWH 135450677 Ki = 189 nM T65200 D03KRW 25192455 IC50 = 1315 nM T65200 D03PVF 16267445 IC50 = 628 nM T65200 D03QYZ 11601544 Ki = 1.4 nM T65200 D04KAZ 44437631 IC50 = 17400 nM T65200 D04LGV 25192457 IC50 = 493 nM T65200 D04WVV 10193044 IC50 = 109 nM T65200 D05ADD 44437632 IC50 = 19600 nM T65200 D05KLE 44160268 IC50 = 10 nM T65200 D05NSB 9450114 IC50 = 200 nM T65200 D06CPL 46890339 IC50 = 820 nM T65200 D06GVN 14314585 IC50 = 9400 nM T65200 D06RKS 11031155 IC50 = 15000 nM T65200 D06UPR 11141268 IC50 = 1310 nM T65200 D07IRZ 44437611 IC50 = 2900 nM T65200 D07LUJ 64945 IC50 = 1900 nM T65200 D08EDV 10893520 IC50 = 5700 nM T65200 D09KDS 4348598 IC50 = 756 nM T65200 D09VPP 21671982 IC50 = 2060 nM T65200 D0A4ZR 135950111 Ki = 10 nM T65200 D0A5JU 52945668 IC50 = 5 nM T65200 D0D3NV 584509 IC50 = 193 nM T65200 D0D3PY 1483443 IC50 = 101 nM T65200 D0DS7W 44237028 IC50 = 117 nM T65200 D0E3ST 3328378 IC50 = 7200 nM T65200 D0EU9W 16750524 IC50 = 60 nM T65200 D0F9RO 6918774 IC50 = 810 nM T65200 D0IO0I 6474893 IC50 = 257 nM T65200 D0J3DW 11850038 IC50 = 16 nM T65200 D0J5RQ 234102 IC50 = 1350 nM T65200 D0J6RQ 6437306 IC50 = 832 nM T65200 D0KG3M 25192460 IC50 = 1069 nM T65200 D0L4VR 636403 Ki = 62 nM T65200 D0L5KQ 135950109 Ki = 1761 nM T65200 D0M3XF 25192606 IC50 = 7 nM T65200 D0M4PP 4271571 IC50 = 75 nM T65200 D0P7RN 1483401 IC50 = 90 nM T65200 D0Q2MI 44437607 IC50 = 1200 nM T65200 D0Q2TF 25192605 IC50 = 466 nM T65200 D0R4DK 46890076 IC50 = 14500 nM T65200 D0T3FW 44419251 IC50 = 64 nM T65200 D0T9NX 44237027 IC50 = 152 nM T65200 D0U8IF 10114 IC50 = 11.3 nM T65200 D0UJ2C 44437618 IC50 = 345 nM T65200 D0V5TC 9111347 IC50 = 291 nM T65200 D0VC2M 2741656 IC50 = 498 nM T65200 D0W9WG 135950108 Ki = 6451 nM T65200 D0Y9XK 46890243 IC50 = 971 nM T65200 D0ZG3Q 135950102 Ki = 4 nM T00872 D0E3TC 44259 IC50 = 0.438 nM T00872 D0O6ZO 9952773 IC50 > 10000 nM T00872 CWM18I 11406175 IC50 > 10000 nM T00872 C1WXC5 11417488 IC50 = 1508 nM T00872 CTG83F 11539329 Ki > 6700 nM T00872 CACS26 11561968 Ki > 2000 nM T00872 CMIL86 11590363 Ki > 6700 nM T00872 C9T6SC 11640926 Ki > 6700 nM T00872 CU0E8O 11690457 Ki > 5000 nM T00872 CFPW41 16007116 Ki > 6700 nM T00872 C7YG1N 24759534 IC50 = 1 nM T00872 CX1HL8 25032704 Ki > 6670 nM T00872 CA51SY 25141108 IC50 < 0.25 nM T00872 C87WKU 25205097 IC50 = 70 nM T00872 CETQ79 44427518 IC50 = 3650 nM T00872 COPG94 44427519 IC50 > 10000 nM T00872 CLI16E 44465026 IC50 = 20 nM T00872 CY3HW5 46224684 IC50 = 210 nM T00872 CLS29B 46872626 IC50 > 10000 nM T00872 C2XTV7 59603828 IC50 = 24 nM T00872 CXJ63M 59603829 IC50 = 6 nM T00872 CQEU96 59603842 IC50 <= 0.5 nM T00872 C09FVB 59603906 IC50 = 1.3 nM T00872 C1M4WZ 59603929 IC50 = 99 nM T00872 CW4QG3 59603981 IC50 = 13 nM T00872 CV63UL 67240318 IC50 > 10000 nM T00872 C9E1NC 68776463 IC50 = 1 nM T00872 CZV54F 68777548 IC50 = 129 nM T00872 C9E8XL 68778264 IC50 = 9 nM T00872 CLR0X7 68779790 IC50 = 43 nM T00872 C5DGR9 69036886 IC50 = 1.2 nM T00872 CPA02V 70841494 IC50 = 5 nM T00872 C1DEQ6 70942743 IC50 = 37 nM T00872 CKT60L 71455860 Ki = 4830 nM T00872 CJ2T9E 76332983 IC50 > 10000 nM T00872 C1HW4B 89735655 IC50 = 5 nM T00872 CH9BP3 127021001 IC50 = 61 nM T00872 C0LY3A 134129875 IC50 = 2100 nM T00872 C6K1TJ 134130033 IC50 = 82 nM T00872 CHV40L 134130103 IC50 = 850 nM T00872 C1Q2AZ 134130107 IC50 = 2564 nM T00872 C7OK6L 134130144 IC50 = 2800 nM T00872 CCW4O0 134130175 IC50 = 226 nM T00872 CDP7Q0 134130181 IC50 = 304 nM T00872 CT5RL6 134130320 IC50 = 60 nM T00872 C12UXV 134130374 IC50 > 30000 nM T00872 C0GRK2 134130397 IC50 = 10 nM T00872 CHQB27 134130448 IC50 = 1524 nM T00872 C18VDQ 134130540 IC50 = 738 nM T00872 CNU0C2 134130690 IC50 = 10 nM T00872 CW3LI4 134130692 IC50 = 80 nM T00872 COX75D 134130730 IC50 = 2800 nM T00872 CJ86AV 134130841 IC50 = 627 nM T00872 CR4TU9 134130878 IC50 = 3000 nM T00872 CM79UL 134130892 IC50 > 30000 nM T00872 C3PR8Q 134130943 IC50 = 14 nM T00872 C08NTZ 134130961 IC50 = 1300 nM T00872 CX51VI 134131112 IC50 = 80 nM T00872 C24LZQ 134131373 IC50 = 1644 nM T00872 C9MXN1 134131388 IC50 = 120 nM T00872 CLG07B 134131413 IC50 = 12770 nM T00872 C02IUK 134131474 IC50 = 4300 nM T00872 CIA49M 134131483 IC50 = 27 nM T00872 CLY29G 134131496 IC50 = 346 nM T00872 CHJ0V1 134131530 IC50 = 1800 nM T00872 CNO5B2 134131560 IC50 = 19 nM T00872 C7YJ0G 155510540 IC50 = 10 nM T00872 C2MD1Q 155513187 IC50 > 10000 nM T00872 C39XGN 155544039 IC50 = 38 nM T00872 CEQO14 155544899 IC50 = 2 nM T00872 CUL01O 155551158 IC50 = 74 nM T00872 CWPX61 155554602 IC50 = 15 nM T00872 CY9N1O 155555954 IC50 = 2.4 nM T00872 C03IWC 155558700 IC50 = 3 nM T00872 CP8HY3 155559157 IC50 = 130 nM T00872 CIGR98 155560320 IC50 = 10 nM T00872 CWCZ68 155562819 IC50 = 9 nM T00872 CI8LZ2 155564791 IC50 = 15 nM T00872 C9OI7A 155568523 IC50 = 22 nM T00872 D00ERW 44444843 Ki > 6667 nM T00872 D00HVA 11624601 Ki > 6700 nM T00872 D03BJF 44465558 IC50 = 12 nM T00872 D0Q3NG 11715520 Ki > 6700 nM T00872 D0S7IE 11658882 Ki > 6700 nM T22956 D0E3TC 44259 IC50 = 6.9 nM T22956 CRC65X 9863786 IC50 > 25000 nM T22956 C3UIL7 44582684 IC50 = 25100 nM T22956 CN4RC3 44582716 IC50 > 100000 nM T22956 CZS9G7 44582745 IC50 = 1220 nM T22956 C9MG0D 44582838 IC50 = 17700 nM T22956 CJ3M5I 134137436 Ki > 1000 nM T22956 CLXN40 155565350 IC50 = 29 nM T53524 D00STL 644241 IC50 < 2.54 nM T53524 D01PZD 5329098 IC50 = 200 nM T53524 D03ZBT 11626560 IC50 > 1000 nM T53524 D04LVK 57379345 IC50 = 1140 nM T53524 D07POC 176870 IC50 = 8120 nM T53524 D08CDI 208908 IC50 > 20000 nM T53524 D0AZ3C 5291 IC50 = 1.995 nM T53524 D0E6XR 3062316 Ki < 10 nM T53524 D0H0EQ 24826799 IC50 = 2.6 nM T53524 D0IQ6P 25102847 IC50 > 10000 nM T53524 D0R0MW 5329102 IC50 = 130 nM T53524 D00DRL 44137946 IC50 < 100 nM T53524 D02UFQ 11620908 IC50 > 10000 nM T53524 D03LWG 53235510 IC50 = 2718 nM T53524 D05PZB 135398495 IC50 = 10 nM T53524 D06KTJ 53252276 IC50 = 45 nM T53524 D07EHV 44814409 IC50 > 10000 nM T53524 D07HPJ 11476171 IC50 = 800 nM T53524 D07HRU 9549295 IC50 = 970 nM T53524 D07KYT 24889392 IC50 = 42 nM T53524 D07PNT 10433653 IC50 = 2 nM T53524 D08HOM 46207586 Ki = 0.7943 nM T53524 D0A5MC 11712649 IC50 = 794.33 nM T53524 D0D1GF 42642645 IC50 = 3.6 nM T53524 D0E3TC 44259 IC50 < 0.1 nM T53524 D0FD6D 11751922 IC50 = 246 nM T53524 D0M0XB 10302451 IC50 = 10000 nM T53524 D0M9QZ 11485656 IC50 = 15 nM T53524 D0O6WV 24794418 IC50 = 28 nM T53524 D0S7HM 16041424 IC50 = 56 nM T53524 D0T2ER 24767976 IC50 = 4.3 nM T53524 D0W7JZ 9911830 IC50 = 2.26 nM T53524 D0T3ME 156422 IC50 > 30000 nM T53524 CB1VW3 1400 IC50 = 657 nM T53524 CWH85P 42723 IC50 = 700 nM T53524 C75EDQ 644355 IC50 = 100 nM T53524 C5HPF3 644356 IC50 = 300 nM T53524 C2DG6J 3068873 IC50 = 2000 nM T53524 CA3C5S 3685259 IC50 < 5000 nM T53524 C9NBG7 5330546 IC50 = 100 nM T53524 CDK3J0 5703619 IC50 = 1.2 nM T53524 C2OL7K 9796455 IC50 = 299 nM T53524 CHF7G5 9890746 IC50 = 210 nM T53524 C3EUB4 9911005 IC50 = 890 nM T53524 CUJR40 10062694 EC50 = 4 nM T53524 CIV15Q 10113978 IC50 = 71 nM T53524 CP95FO 10181075 IC50 = 139 nM T53524 CSGD16 10246246 IC50 > 7000 nM T53524 C95LYF 10457505 IC50 = 710 nM T53524 CJ4P5T 10905857 IC50 = 770 nM T53524 CJ05CL 11048367 IC50 = 90 nM T53524 CR2O3F 11155047 IC50 = 3.6 nM T53524 C84NJO 11155950 IC50 = 43 nM T53524 CIA1Q6 11167070 IC50 = 17 nM T53524 CP4GL8 11212549 IC50 = 3.3 nM T53524 CT7X1E 11213083 IC50 = 10 nM T53524 CY2PF1 11224592 IC50 = 5.8 nM T53524 C06FWR 11224992 IC50 = 14 nM T53524 CW94ZU 11225456 IC50 = 37 nM T53524 C9CGI8 11225457 IC50 < 10 nM T53524 CFJ0W9 11236257 IC50 = 52 nM T53524 CFJ2C0 11236308 IC50 = 3.5 nM T53524 C8S2HR 11237059 IC50 = 24 nM T53524 C4R2CE 11247801 IC50 = 2 nM T53524 C71ONE 11259460 IC50 = 24 nM T53524 CLE31R 11259708 IC50 = 18 nM T53524 CPI45C 11270447 IC50 = 5.8 nM T53524 CMZ49B 11270888 IC50 = 1.6 nM T53524 CUO27S 11282791 IC50 = 17 nM T53524 CC9OM5 11292923 IC50 = 3.6 nM T53524 CHKY86 11305057 IC50 = 3.9 nM T53524 CHQ6O9 11316725 IC50 = 21 nM T53524 CLX54H 11317348 IC50 = 67 nM T53524 C2MY9F 11327849 IC50 = 3.6 nM T53524 C9GI6J 11328439 IC50 = 3.4 nM T53524 C9BZ5Q 11339914 IC50 = 4.7 nM T53524 C4VB3D 11339915 IC50 = 6.8 nM T53524 CI6ZX5 11350985 IC50 = 6.4 nM T53524 C12LUM 11352232 IC50 < 3 nM T53524 CL4Z7M 11374372 IC50 = 10 nM T53524 C0S1OV 11385268 IC50 = 2 nM T53524 CJUC63 11409093 IC50 = 75 nM T53524 CXH8R6 11441787 IC50 = 36 nM T53524 C60VOM 11443129 IC50 = 13 nM T53524 C1U4GO 11465344 IC50 = 6.8 nM T53524 CI59ZS 11488585 IC50 = 55 nM T53524 CRJ3H2 11495362 IC50 = 5 nM T53524 CMIT06 11496035 IC50 = 46 nM T53524 C9DV1X 11525218 IC50 = 6 nM T53524 C98ENG 11525727 IC50 = 28 nM T53524 CL7X4Q 11530963 IC50 = 943 nM T53524 COJI59 11539040 IC50 = 12 nM T53524 CACS26 11561968 Ki > 2000 nM T53524 C9CDX4 11583287 IC50 = 37 nM T53524 CI5W0C 11583439 IC50 = 8 nM T53524 CQ5NP2 11604829 IC50 = 9 nM T53524 CFM2Y4 11640405 IC50 = 7 nM T53524 C08DMH 11655667 IC50 = 15 nM T53524 CO52CP 11656170 IC50 = 5 nM T53524 CG5PS9 11685945 IC50 = 62 nM T53524 CU0E8O 11690457 Ki > 10000 nM T53524 C2CM0L 11690679 IC50 = 40 nM T53524 CSIN39 11690947 IC50 = 18 nM T53524 CB0AP2 11705863 Ki > 10000 nM T53524 C45EWD 11723489 IC50 = 300 nM T53524 C9P0VD 11729539 IC50 = 240 nM T53524 C8EB4Y 11775063 Ki = 2.512 nM T53524 CDZ1I3 11989153 IC50 = 406 nM T53524 C3YRU7 15295578 IC50 = 40500 nM T53524 C7LB4I 15949613 IC50 = 35 nM T53524 C9TU1O 16046126 IC50 > 1000 nM T53524 C5VPH9 16129448 IC50 = 4310 nM T53524 CI62OL 18451141 Ki > 10000 nM T53524 CL81VC 21100709 IC50 = 4040 nM T53524 C6JV7W 23400934 IC50 > 7000 nM T53524 CD5S7O 23401001 IC50 > 7000 nM T53524 CI6C1R 23658582 IC50 = 4 nM T53524 C2RV3U 24180608 IC50 > 30000 nM T53524 CJL67N 24759089 IC50 = 3 nM T53524 CAJ4T2 24762205 IC50 = 74 nM T53524 C2UOE0 24766030 IC50 > 50000 nM T53524 CW0G8H 24812719 IC50 = 9 nM T53524 C43HWQ 24883287 IC50 > 10000 nM T53524 C8DA5Q 24883334 IC50 > 10000 nM T53524 C2ICS7 25065806 IC50 = 221 nM T53524 CTV54O 25123227 IC50 = 12 nM T53524 CLFM35 25206064 IC50 = 44000 nM T53524 C6FGQ1 25206346 IC50 = 43 nM T53524 CNQ9G5 25218180 IC50 < 1000 nM T53524 CLW80F 44160269 IC50 = 10000 nM T53524 CK73NR 44219749 IC50 > 50000 nM T53524 CEL61X 44229839 IC50 > 10000 nM T53524 CX6YU4 44388576 IC50 = 490 nM T53524 C74BAO 44409484 IC50 = 6 nM T53524 C5OK1I 44409504 IC50 = 4 nM T53524 C8W5YG 44447872 IC50 = 69 nM T53524 C4WRN5 44541014 IC50 = 50000 nM T53524 CCL85F 44575073 IC50 > 50000 nM T53524 CJX06P 44575126 IC50 = 27100 nM T53524 CE8FC7 44575127 IC50 = 36200 nM T53524 C9VXN3 44578709 IC50 > 10000 nM T53524 C28QLM 44605035 IC50 > 50000 nM T53524 C75XHS 44605037 IC50 > 50000 nM T53524 CC95PQ 45375865 IC50 > 50000 nM T53524 CEOQ27 45375866 IC50 > 50000 nM T53524 C4KWJ3 45379956 IC50 > 100000 nM T53524 C2CU0B 45380067 IC50 = 26170 nM T53524 C6E2SC 45482700 IC50 > 10000 nM T53524 CZXH74 45482750 IC50 > 10000 nM T53524 C96BNW 46179972 IC50 = 38 nM T53524 CF57GK 46215462 IC50 = 20 nM T53524 C2P9QO 46228508 IC50 = 1840 nM T53524 C6E5PY 46228822 IC50 = 9710 nM T53524 C3T8AM 46228951 IC50 = 2170 nM T53524 CYZV41 46231219 IC50 = 1800 nM T53524 C7J5UP 46231220 IC50 = 1307 nM T53524 CC96GZ 46231221 IC50 = 1156 nM T53524 CO3P0J 46866604 IC50 < 50000 nM T53524 C5WC9K 46871765 IC50 = 3000 nM T53524 CJOM49 46880136 IC50 = 6560 nM T53524 CTZ71Y 46898039 IC50 = 0.98 nM T53524 C2B5XF 49765254 IC50 > 10000 nM T53524 CHSF07 49806372 IC50 > 1000 nM T53524 CJ3SU6 49830359 Ki = 50.12 nM T53524 CBCF39 49830372 Ki > 10000 nM T53524 CJZ5A0 49840306 IC50 > 10000 nM T53524 CB0S2P 49842666 IC50 = 27 nM T53524 C5R6QY 49842669 IC50 = 1200 nM T53524 C0NA9U 49842670 IC50 = 87 nM T53524 CC7MR2 49842671 IC50 = 1400 nM T53524 CAI20B 49842778 IC50 = 89 nM T53524 CRA74I 49842779 IC50 = 95 nM T53524 CS9G6E 50997096 IC50 > 10000 nM T53524 CB9C8G 51351016 IC50 = 1540 nM T53524 COD9Y2 51351017 IC50 = 1080 nM T53524 CW96FU 51351018 IC50 = 4890 nM T53524 CR9T2E 51351019 IC50 = 4110 nM T53524 CEQN27 52936621 Ki > 1000 nM T53524 C6L8WI 52945628 IC50 = 67 nM T53524 C8ZTF9 53249002 IC50 = 295 nM T53524 C09SDH 53257410 IC50 > 10000 nM T53524 C2P3OT 53316977 IC50 = 2300 nM T53524 CZ0BV7 53320342 IC50 = 180 nM T53524 CX59LD 53320915 IC50 = 8600 nM T53524 CZY0J7 53323592 IC50 = 450 nM T53524 C2W9OA 53324451 IC50 = 7.23 nM T53524 CCKD48 53324892 IC50 = 14000 nM T53524 CNPM14 53341082 IC50 > 3000 nM T53524 CBK9Q6 53357848 IC50 > 10000 nM T53524 C8NA4L 53384644 IC50 > 30000 nM T53524 C0SC3J 54672928 IC50 = 85 nM T53524 CDMS75 54672929 IC50 = 52 nM T53524 CP5ZC3 54672931 IC50 = 104 nM T53524 C6OS4F 54672932 IC50 = 94 nM T53524 CR64QL 54673093 IC50 = 80 nM T53524 CE1D2H 54673094 IC50 = 97 nM T53524 CJL9T7 54673095 IC50 = 130 nM T53524 C73LSR 54673096 IC50 = 96 nM T53524 CBO2L1 54761157 IC50 = 6.2 nM T53524 CS23GM 54762055 IC50 = 9.2 nM T53524 CFJ37O 56649380 IC50 = 86 nM T53524 CV8B1X 56649401 IC50 = 95 nM T53524 CUEW30 56649402 IC50 = 75 nM T53524 CK2OT6 56649403 IC50 = 72 nM T53524 CVN1Z8 56649405 IC50 = 140 nM T53524 CR50TJ 56835147 IC50 = 1355 nM T53524 C87YOZ 56929808 IC50 = 8 nM T53524 C9MJG4 56929824 IC50 = 860 nM T53524 CCW89V 56932477 IC50 = 1187 nM T53524 CR3FK5 56932525 IC50 = 11.8 nM T53524 C0YO5U 56932528 IC50 = 245 nM T53524 CI6QE5 56970263 IC50 < 500 nM T53524 C62OJE 56970264 IC50 = 150 nM T53524 CZSM95 57412684 IC50 > 10000 nM T53524 C8P6RD 57505528 IC50 = 13 nM T53524 C8R4FE 57991377 IC50 = 546.7 nM T53524 CH7L5N 58172700 IC50 = 8.2 nM T53524 CP34RY 59394193 IC50 = 150 nM T53524 C1MR8Q 60097495 IC50 > 10000 nM T53524 C9ZCT2 62705065 IC50 > 1000 nM T53524 C1HSE0 67035086 IC50 = 900 nM T53524 CWI6K5 67035106 IC50 > 10000 nM T53524 C38RGB 67035556 IC50 > 10000 nM T53524 C37NKO 67129970 IC50 > 10000 nM T53524 CK80LJ 67130050 IC50 > 10000 nM T53524 CQ97ZW 67161103 IC50 = 20 nM T53524 CNP52W 67163022 IC50 = 6 nM T53524 CV63UL 67240318 IC50 > 10000 nM T53524 C8I7GC 68293638 IC50 = 5300 nM T53524 CD56XK 68293660 IC50 > 10000 nM T53524 C7GRV2 68755406 IC50 > 10000 nM T53524 C0HA8V 68783839 IC50 = 1 nM T53524 CAIO65 68796885 IC50 = 50 nM T53524 CH6S7Q 70681377 Ki > 10000 nM T53524 C48ZLN 71060894 IC50 = 22 nM T53524 C10CHQ 71060955 IC50 = 127 nM T53524 CWO0S3 71061505 IC50 = 54 nM T53524 CZD6W0 71283030 IC50 = 1.3 nM T53524 CT1NU9 71283192 IC50 = 0.18 nM T53524 CL6B7O 71283325 IC50 = 0.75 nM T53524 CR05MO 71283371 IC50 = 1.2 nM T53524 CHX4F3 71283395 IC50 = 0.19 nM T53524 COR61Q 71283495 IC50 = 0.96 nM T53524 CI27GT 71283528 IC50 = 3.2 nM T53524 CD8LZ0 71283574 IC50 = 0.32 nM T53524 C8OGT4 71283628 IC50 = 0.2 nM T53524 C6A5JN 71291191 IC50 = 0.09 nM T53524 CEBO91 71452977 IC50 > 10000 nM T53524 CQY31T 71498139 IC50 = 27.3 nM T53524 C9DIK2 71512060 IC50 = 3596 nM T53524 C6HF8S 71521082 IC50 = 83.87 nM T53524 C9Z3AI 71521083 IC50 = 25.96 nM T53524 CRX81Q 71575642 IC50 = 223 nM T53524 C1BCX0 71579696 IC50 > 1000 nM T53524 CZ31PU 71583657 IC50 > 10000 nM T53524 C1FAU8 71679855 IC50 = 390 nM T53524 C3OS8U 71714087 IC50 = 120 nM T53524 C92AZQ 71714088 IC50 = 250 nM T53524 CN1Y9I 71714230 IC50 = 540 nM T53524 CM6NE9 71714231 IC50 = 60 nM T53524 CG28AP 71714232 IC50 = 150 nM T53524 C67HDT 71714234 IC50 = 46 nM T53524 CRS05F 71714235 IC50 = 13 nM T53524 CVC19T 71714373 IC50 = 91 nM T53524 CD5C8J 71714374 IC50 = 1700 nM T53524 C51ISR 71714375 IC50 = 60 nM T53524 C5HJK2 71714376 IC50 < 3 nM T53524 C70SJV 71714377 IC50 = 31 nM T53524 CKNB62 71720020 IC50 = 262 nM T53524 CU1IL6 71741204 IC50 > 100000 nM T53524 CN1GA3 71741327 IC50 > 100000 nM T53524 COS5D7 71741328 IC50 > 100000 nM T53524 C8PWZ0 71741329 IC50 > 100000 nM T53524 CT4XR9 71741332 IC50 > 50000 nM T53524 C4Q6FE 71815105 IC50 = 7.2 nM T53524 C60TUV 72737208 IC50 > 10000 nM T53524 CJ3WA6 72737404 IC50 > 10000 nM T53524 C2PAK9 73438493 IC50 = 1280 nM T53524 CBAT06 76071144 IC50 = 672 nM T53524 CH8W7D 77461036 IC50 > 1000 nM T53524 CCJ43A 86302281 IC50 > 10000 nM T53524 CB5NJ4 86302541 IC50 = 548.6 nM T53524 CPG3A5 86302574 IC50 > 30000 nM T53524 CX29IY 90655145 IC50 > 10000 nM T53524 CK72FW 102129497 IC50 = 15.73 nM T53524 CTGP06 117996541 IC50 > 10000 nM T53524 C2IN3C 118710236 IC50 < 1 nM T53524 CF2YR1 118710237 IC50 < 1 nM T53524 CQCX41 118737057 IC50 = 890 nM T53524 C8U0ZH 118737468 IC50 = 3.26 nM T53524 C75PHN 119058124 IC50 = 420 nM T53524 CKBP72 121231408 IC50 > 10000 nM T53524 C81IFQ 122163152 IC50 > 100000 nM T53524 C4X7SD 122192466 IC50 = 370 nM T53524 CD67LU 122705248 IC50 > 10000 nM T53524 CX63VW 122705258 IC50 > 10000 nM T53524 C76IKM 122705261 IC50 > 10000 nM T53524 CY30FL 123752658 IC50 = 5.6 nM T53524 C8ALO2 124088839 IC50 > 10000 nM T53524 C8KXV1 127025843 IC50 > 1000 nM T53524 CKS28E 127034802 IC50 = 402 nM T53524 CKX40V 127037812 IC50 = 106.8 nM T53524 C70RUP 127038480 IC50 > 10000 nM T53524 C3WCN8 127041777 IC50 = 19.6 nM T53524 CG8DA9 127045861 IC50 > 100000 nM T53524 CC4ND8 127046862 IC50 > 100000 nM T53524 CO25WH 127052538 IC50 > 10000 nM T53524 CF5D2Y 129318936 IC50 = 132 nM T53524 C0FM1R 130196825 IC50 = 970 nM T53524 CUO0C5 132156633 IC50 > 10000 nM T53524 C6OMB1 132204257 IC50 = 426 nM T53524 CJ04HZ 132585195 IC50 = 7.2 nM T53524 C53OJM 132607333 IC50 = 19.13 nM T53524 CERS64 132937256 IC50 = 27606 nM T53524 CM06HV 133081975 IC50 = 27 nM T53524 CQ5SI2 134135403 IC50 = 1.6 nM T53524 C5BDS1 134144754 IC50 = 1.3 nM T53524 CN35SO 134146628 IC50 > 1000 nM T53524 CUKE45 134147919 IC50 = 95.23 nM T53524 C5JSP7 134151944 IC50 = 0.53 nM T53524 CBK9O8 134153891 IC50 = 13 nM T53524 CVTN56 134156672 IC50 < 0.1 nM T53524 C2AN7T 134611886 IC50 > 100000 nM T53524 CYL5V1 134694986 IC50 = 2357 nM T53524 C76JPR 135405015 IC50 = 3 nM T53524 CV8Q7A 135430397 IC50 = 6 nM T53524 CS63IO 135476717 IC50 = 59 nM T53524 CA80OZ 135488014 IC50 = 7 nM T53524 CDCF48 135488027 IC50 = 7 nM T53524 CG5HY4 135507297 IC50 = 5 nM T53524 CT0NV5 135514617 IC50 = 17 nM T53524 CFPV27 135543821 IC50 = 10 nM T53524 CRCH86 135546221 IC50 = 431 nM T53524 C65XMQ 135546228 IC50 = 6 nM T53524 CPHG43 135567142 IC50 = 9 nM T53524 CJ7U4C 136053657 IC50 = 212.3 nM T53524 CU05YS 136118622 IC50 = 13 nM T53524 CN49OS 136118623 IC50 = 55 nM T53524 CR48NF 136118625 IC50 = 844 nM T53524 CD5M9T 136118626 IC50 = 614 nM T53524 CW27AO 136118641 IC50 = 1950 nM T53524 CDT7E4 136211077 IC50 = 781.8 nM T53524 CE7L0G 136269119 IC50 > 50000 nM T53524 C7U9GP 136269138 IC50 > 50000 nM T53524 CCM42D 137249694 IC50 = 6.6 nM T53524 C25ERN 137631967 IC50 > 100 nM T53524 CV49KX 137632804 IC50 = 106 nM T53524 CE1B7Y 137633677 IC50 = 262 nM T53524 CMY81W 137633944 IC50 = 127 nM T53524 CNX0F9 137634126 IC50 = 74 nM T53524 CI1E8V 137634241 IC50 = 5590 nM T53524 CPFH76 137634323 IC50 = 1465 nM T53524 CILC91 137635352 IC50 = 83 nM T53524 CBP52G 137635849 IC50 = 32 nM T53524 CK8G2R 137636007 IC50 = 83 nM T53524 CEL8G1 137636465 IC50 = 164 nM T53524 CL1Q8V 137637006 IC50 = 305 nM T53524 C06JRX 137637094 IC50 > 100 nM T53524 CLFR07 137637309 IC50 = 928 nM T53524 CP2B8Y 137639044 IC50 > 50000 nM T53524 CI7WH5 137639132 IC50 = 157 nM T53524 CI5K8B 137640242 IC50 = 124 nM T53524 CA70ZG 137641063 IC50 = 136 nM T53524 CW3C1G 137641107 IC50 = 22 nM T53524 CO18WK 137641971 IC50 = 576 nM T53524 C52EZY 137642247 IC50 = 1081 nM T53524 CJ4S0F 137642960 IC50 = 1779 nM T53524 CVF3Y4 137643942 IC50 = 65 nM T53524 C9F6VM 137645016 IC50 = 401 nM T53524 C2BP8R 137645569 IC50 = 87 nM T53524 CF92BJ 137646079 IC50 = 18925 nM T53524 C5B7PN 137647552 IC50 = 309 nM T53524 C0E5LD 137647791 IC50 = 43877 nM T53524 CITB67 137647879 IC50 > 5000 nM T53524 C8CYG9 137648008 IC50 = 411 nM T53524 CGI1F8 137649216 IC50 = 135 nM T53524 CTF9N6 137649662 IC50 = 27 nM T53524 CVK6O2 137650604 IC50 = 21400 nM T53524 CI6X0A 137651311 IC50 = 137 nM T53524 CIM42E 137651341 IC50 = 87 nM T53524 C1DK0P 137651391 IC50 > 100 nM T53524 CL2GW4 137652151 IC50 = 387 nM T53524 C28QUP 137652864 IC50 > 10000 nM T53524 CHP3E8 137653224 IC50 = 472 nM T53524 CZS0M4 137653919 IC50 = 22 nM T53524 C78DVY 137654650 IC50 = 1179 nM T53524 CS21QO 137654848 IC50 > 50000 nM T53524 CIS4O3 137655297 IC50 = 182 nM T53524 C9ZIV1 137655363 IC50 = 176 nM T53524 C17LIA 137655641 IC50 = 174.6 nM T53524 CQ70VE 137655849 IC50 > 50000 nM T53524 C0RQB3 137656341 IC50 = 1133 nM T53524 CZ4C1M 137656917 IC50 = 313 nM T53524 CO61JG 137657076 IC50 = 732 nM T53524 CV9H6B 137657843 IC50 = 4608 nM T53524 CV5H3Z 137657932 IC50 > 100 nM T53524 C98AVI 137657952 IC50 > 5000 nM T53524 CPV1S9 137658287 IC50 = 172 nM T53524 C81LTC 137658404 IC50 = 215 nM T53524 CQMB10 137658515 IC50 = 40 nM T53524 CX53JP 137658925 IC50 = 1123 nM T53524 C4FKX3 137659066 IC50 = 1101 nM T53524 CKVS16 137659546 IC50 = 97 nM T53524 C8D9NE 137660511 IC50 = 560 nM T53524 CM5T3L 137660584 IC50 > 50000 nM T53524 C7FZA8 137660733 IC50 = 4077 nM T53524 C8WZ2V 137661264 IC50 = 1572 nM T53524 C09NZL 137661683 IC50 = 82 nM T53524 CHB9P7 137661707 IC50 = 24 nM T53524 C07EKN 138454794 IC50 = 7777 nM T53524 CUXO19 138617501 IC50 > 1000 nM T53524 C6AK0N 139030518 IC50 = 25 nM T53524 CS9Z4A 141523058 IC50 > 50000 nM T53524 CUV1P6 141523059 IC50 > 50000 nM T53524 C2CZ1Q 141523061 IC50 > 50000 nM T53524 C98TNO 141523067 IC50 > 50000 nM T53524 CJQC54 141523068 IC50 > 50000 nM T53524 CW47GO 141523069 IC50 > 50000 nM T53524 CUV07Y 141523072 IC50 = 7500 nM T53524 CKBQ94 141523076 IC50 > 50000 nM T53524 C4ASE6 141523085 IC50 > 50000 nM T53524 CT37IP 141523091 IC50 > 50000 nM T53524 C4LA8F 141523094 IC50 > 50000 nM T53524 C34CKN 141523354 IC50 = 4.35 nM T53524 C1IX5N 145956333 IC50 = 4.4 nM T53524 C7W4JR 145964096 IC50 = 66 nM T53524 CWJ8Z5 145964314 IC50 = 96 nM T53524 CCX9I4 145964954 IC50 = 1412 nM T53524 C2BV7H 145964972 IC50 = 60 nM T53524 CZV30K 145965543 IC50 = 188 nM T53524 CF4N6D 145966189 IC50 = 290 nM T53524 CMNO25 145966658 IC50 = 1233 nM T53524 CQE9M5 145966810 IC50 = 990 nM T53524 CRE5N6 145968259 IC50 = 195 nM T53524 CW65FJ 145968494 IC50 = 5099 nM T53524 CNT9I4 145968729 IC50 > 20000 nM T53524 CWJ12M 145969155 IC50 = 370 nM T53524 CMD17C 145969392 IC50 = 59 nM T53524 C29CWG 145971794 IC50 = 156 nM T53524 CEX15Q 145971884 IC50 = 1090 nM T53524 CS9PM6 145972964 IC50 = 1031 nM T53524 CSO3Y9 145973328 IC50 = 35 nM T53524 CI7S1H 145973461 IC50 = 1496 nM T53524 C95UKI 145974361 IC50 = 150 nM T53524 CD5FC2 145974374 IC50 = 7655 nM T53524 CJ46RB 145975271 IC50 = 160 nM T53524 C74TYP 145975351 IC50 = 691.5 nM T53524 CXW3I9 145975391 IC50 > 20000 nM T53524 C0I6RX 145975438 IC50 = 154 nM T53524 CH3UR1 145975624 IC50 = 66 nM T53524 CZ86GY 145976023 IC50 = 4739 nM T53524 CP6I4J 145978173 IC50 = 3197 nM T53524 CQG83B 145978348 IC50 = 452 nM T53524 CZC8M4 145978823 IC50 = 187 nM T53524 CUNA14 145983151 IC50 > 50000 nM T53524 CD39VL 145983968 IC50 = 2200 nM T53524 C3L9WK 145984021 IC50 = 28100 nM T53524 C35ABX 155512081 IC50 = 1849 nM T53524 C1NLI6 155512420 IC50 = 1248 nM T53524 C2MD1Q 155513187 IC50 > 10000 nM T53524 C8FLN7 155515952 IC50 = 37 nM T53524 C8RH7M 155516997 IC50 = 7 nM T53524 C4JH8L 155517052 IC50 = 11 nM T53524 C7XZD8 155517171 IC50 = 167 nM T53524 C0X1QH 155517531 IC50 = 236 nM T53524 C86HPW 155518524 IC50 = 48000 nM T53524 COZW68 155519778 IC50 = 211 nM T53524 CL4HE2 155521618 IC50 = 686 nM T53524 C72JXV 155523168 IC50 = 1351 nM T53524 CXFH76 155523422 IC50 = 644 nM T53524 CNL1D3 155524029 IC50 = 1024 nM T53524 CV8GU5 155525848 IC50 = 1813 nM T53524 CFL79R 155526188 IC50 = 47 nM T53524 CLFK05 155527869 IC50 = 1292 nM T53524 CPZ5H2 155529814 IC50 = 118 nM T53524 CA1F3X 155532001 IC50 = 121 nM T53524 CZ39MW 155534364 IC50 = 47 nM T53524 C3LC9I 155536820 IC50 = 3644 nM T53524 C76UDB 155537564 IC50 = 65 nM T53524 CA7ZV6 155539272 IC50 = 26 nM T53524 C8EIL4 155539972 IC50 = 128 nM T53524 CE46SL 155540854 IC50 > 30000 nM T53524 C5O4JM 155540856 IC50 > 30000 nM T53524 CE0AS9 155541726 IC50 = 1131 nM T53524 C3GW4A 155545834 IC50 = 36 nM T53524 C0YC4S 155546245 IC50 = 156 nM T53524 C7SF2C 155547229 IC50 = 242 nM T53524 CF53LM 155548191 IC50 = 39 nM T53524 CN90LV 155549976 IC50 = 14 nM T53524 CJNH17 155552580 IC50 = 25 nM T53524 CN3G6E 155553739 IC50 = 6 nM T53524 C3N6XG 155554070 IC50 > 20000 nM T53524 CGVU70 155554426 IC50 > 30000 nM T53524 C7OKM0 155555183 IC50 = 33 nM T53524 C4OA5Y 155556204 IC50 = 35 nM T53524 CD1MJ8 155557135 IC50 > 20000 nM T53524 C0WS3K 155557668 IC50 = 5 nM T53524 C03EYH 155559593 IC50 = 74 nM T53524 C0C1UI 155559734 IC50 = 182 nM T53524 C8WUE3 155559832 IC50 = 94 nM T53524 C3ZP6O 155564128 IC50 = 73 nM T53524 C8ZIP2 155564344 IC50 > 20000 nM T53524 C8MU1I 155564722 IC50 = 32 nM T53524 C94IJB 10367131 IC50 = 3 nM T53524 CI8LX0 57976125 IC50 = 5 nM T53524 D01YWE 25207521 IC50 = 11100 nM T53524 D02BXJ 46864270 IC50 = 1.3 nM T53524 D05FFB 91643 IC50 = 600 nM T53524 D06HVH 54613583 IC50 > 10000 nM T53524 D0BW4G 10907042 IC50 = 50 nM T53524 D0C2GE 67161540 IC50 = 3 nM T53524 D0D2FC 2794188 IC50 > 20000 nM T53524 D0Q4EQ 16742063 IC50 = 1110 nM T53524 D0R2WK 16038120 EC50 > 1000 nM T53524 D0U3NI 53246941 IC50 = 956 nM T53524 D0V4EX 54760053 IC50 = 7.7 nM T53524 D0XS9E 5330535 IC50 = 1000 nM T53524 D0YZ7H 9797370 IC50 = 45 nM T10965 D02AUB 9811353 IC50 = 70000 nM T10965 D0Z0AM 12004316 IC50 = 125000 nM T10965 C4AC2Z 159321 IC50 = 5000 nM T10965 C1GDY7 587790 IC50 = 31800 nM T10965 C96KNY 643990 IC50 > 1000000 nM T10965 CME97N 9852751 IC50 = 50000 nM T10965 CZ98HT 9977686 IC50 > 500000 nM T10965 C8TZ5Q 10101726 IC50 = 290 nM T10965 C2VX3P 10886395 IC50 = 17000 nM T10965 CA7R6X 10896694 IC50 = 21000 nM T10965 C73NDA 10941391 IC50 = 100000 nM T10965 CN4S3X 11060508 IC50 = 16000 nM T10965 CWL2J0 11152028 IC50 = 250000 nM T10965 CJ02YL 11153082 IC50 = 1250000 nM T10965 CVU83H 11153727 IC50 = 550000 nM T10965 CR3YS9 11188155 IC50 = 150000 nM T10965 C6VYS0 11201127 IC50 = 10000000 nM T10965 CT2L8I 11210832 IC50 = 138000 nM T10965 CR3TS0 11222068 IC50 = 500000 nM T10965 C5WBN7 11223255 IC50 <= 6000 nM T10965 CB9OA0 11225060 IC50 <= 2000 nM T10965 COL58J 11232405 IC50 = 550000 nM T10965 C16VKQ 11234111 IC50 = 225000 nM T10965 CNL6D9 11234390 IC50 = 325000 nM T10965 CST70G 11236859 IC50 = 500000 nM T10965 C8AFW9 11244687 IC50 = 413000 nM T10965 CKW1R0 11248935 IC50 <= 4000 nM T10965 C4Z0FP 11258464 IC50 = 10200 nM T10965 CV7MP0 11280717 IC50 = 100000 nM T10965 C3P7QJ 11293661 IC50 <= 10000 nM T10965 C1OT9D 11315434 IC50 = 225000 nM T10965 CM8YN2 11348172 IC50 = 413000 nM T10965 C2AL9B 11359737 IC50 = 475000 nM T10965 C76IZB 11359995 IC50 = 450000 nM T10965 C5F1EZ 11383708 IC50 = 200000 nM T10965 CA0ZP8 11405964 IC50 = 123000 nM T10965 C4H8DK 11418639 IC50 = 610000 nM T10965 C7S8HV 11453647 IC50 = 625000 nM T10965 CR5UW7 11463943 IC50 <= 6000 nM T10965 C48AGV 11486189 IC50 = 425000 nM T10965 CKHO40 11558561 IC50 = 19000000 nM T10965 CN5M7E 11680708 IC50 = 19500000 nM T10965 CN92PV 11738934 IC50 = 1000000 nM T10965 CD6T9P 11773900 IC50 <= 6000 nM T10965 CB72VE 11785253 IC50 <= 2000 nM T10965 CR6W3S 16099936 IC50 = 1500000 nM T10965 CXI6J0 16100062 IC50 = 225000 nM T10965 C1NBI3 16100075 IC50 = 200000 nM T10965 C0VW7M 16100078 IC50 = 225000 nM T10965 C51UWL 16100080 IC50 = 175000 nM T10965 C2NO7U 16100082 IC50 = 175000 nM T10965 C6OXK4 16100084 IC50 = 200000 nM T10965 CU0O3W 16100086 IC50 = 400000 nM T10965 CG2CI3 16100088 IC50 = 270000 nM T10965 CR5PW2 16100092 IC50 = 545000 nM T10965 C30LWH 16100094 IC50 = 175000 nM T10965 C3LUQ9 16100095 IC50 = 190000 nM T10965 C8BOR2 16100096 IC50 = 175000 nM T10965 C76FWX 16100097 IC50 = 400000 nM T10965 CXK19G 16100098 IC50 = 250000 nM T10965 C29XLR 16100099 IC50 = 390000 nM T10965 C9RYJ6 16100104 IC50 = 225000 nM T10965 C4ZXU1 16100107 IC50 = 650000 nM T10965 C82QOH 16100109 IC50 = 415000 nM T10965 CEW9U4 16100113 IC50 = 250000 nM T10965 CEQJ37 16100148 IC50 = 300000 nM T10965 C5BZ4G 16100154 IC50 = 715000 nM T10965 CA9MZ5 16100159 IC50 = 900000 nM T10965 C9E1DO 16100168 IC50 = 380000 nM T10965 CHU54W 16100189 IC50 = 125000 nM T10965 C20KGX 16100199 IC50 = 580000 nM T10965 C62DAO 16114614 IC50 = 1100 nM T10965 C1ET3V 16114615 IC50 = 2100 nM T10965 CQ90BS 16114616 IC50 = 2400 nM T10965 CA4MJ7 16114618 IC50 = 34900 nM T10965 CWGO19 16114619 IC50 = 2900 nM T10965 CTC76N 16114620 IC50 = 21700 nM T10965 CM7Z2R 16115893 IC50 = 870 nM T10965 C41WNZ 16116039 IC50 = 4200 nM T10965 CUE4D8 16116040 IC50 = 43200 nM T10965 C2EHS8 16116042 IC50 = 19600 nM T10965 CTG1J6 16116159 IC50 = 2300 nM T10965 CZH0G1 16116162 IC50 = 14800 nM T10965 C5GZB3 16116163 IC50 = 42800 nM T10965 CG05BP 16116164 IC50 > 500000 nM T10965 CKI2E4 16116165 IC50 = 53900 nM T10965 C5Q4GR 16116166 IC50 = 28600 nM T10965 C7F1DY 16116286 IC50 = 19500 nM T10965 CU4OF0 16116421 IC50 = 57200 nM T10965 C89WXF 16116422 IC50 = 7600 nM T10965 C82KGR 16116555 IC50 = 24800 nM T10965 C9DME7 16116556 IC50 = 3400 nM T10965 CU2IB8 16116557 IC50 = 5800 nM T10965 CTXB17 16116558 IC50 = 21800 nM T10965 CFU0D9 16116559 IC50 = 212100 nM T10965 C7WJ0Y 16725848 IC50 = 570 nM T10965 CC12EZ 23709469 IC50 = 100000 nM T10965 C4DEG9 44264802 IC50 = 500 nM T10965 CQP9G7 44304820 IC50 = 300000 nM T10965 C5PC9B 44314807 IC50 = 41000 nM T10965 C8V5HM 44314808 IC50 = 127000 nM T10965 C9YI8T 44314810 IC50 = 7000 nM T10965 C9FOU7 44314839 IC50 = 1000 nM T10965 C4FE2A 44314950 IC50 = 15000 nM T10965 CMR6V4 44314968 IC50 = 28000 nM T10965 C7S8PZ 44314993 IC50 = 87000 nM T10965 CG2R9Y 44314996 IC50 = 85000 nM T10965 CH5N4J 44315249 IC50 = 25000 nM T10965 CZ06IY 44315261 IC50 = 39000 nM T10965 CJN5S6 44315290 IC50 = 28000 nM T10965 CE18QO 44315291 IC50 = 76000 nM T10965 C7J8LN 44315330 IC50 = 4000 nM T10965 CECK48 44315332 IC50 = 20000 nM T10965 C30ZLU 44315665 IC50 = 10600 nM T10965 CUIE94 44339430 IC50 > 50000 nM T10965 C0CI4Z 44339486 IC50 = 640 nM T10965 CD1Y6W 44340382 IC50 = 40000 nM T10965 CC7G9J 44340394 IC50 = 5000 nM T10965 C2Q7LW 44340567 IC50 = 1000 nM T10965 CZG4T2 44340638 IC50 = 8000 nM T10965 CK1GA0 44340639 IC50 = 3000 nM T10965 CICW90 44356343 IC50 = 15000 nM T10965 C1VH5G 44356439 IC50 = 3600 nM T10965 CK7WE9 44356515 IC50 = 37000 nM T10965 CPM04F 44356616 IC50 = 1600 nM T10965 C8CR4F 44356617 IC50 = 250000 nM T10965 CXL0S8 44387278 IC50 > 1000000 nM T10965 CIAL79 44387290 IC50 = 44000 nM T10965 CHIF62 44387291 IC50 > 1000000 nM T10965 C6FK5A 44387293 IC50 > 1000000 nM T10965 C7WPK9 44387294 IC50 > 1000000 nM T10965 CPQ09T 44387295 IC50 = 670000 nM T10965 CPT5K3 44387297 IC50 = 560000 nM T10965 CDUL51 44398683 IC50 <= 3000 nM T10965 CQH4D1 44398719 IC50 <= 2000 nM T10965 C2Z1PN 44398755 IC50 <= 2000 nM T10965 CS0M3D 44399068 IC50 = 40000000 nM T10965 C67QAL 44399069 IC50 > 50000000 nM T10965 C3TJ5S 44399147 IC50 > 50000000 nM T10965 CB74WV 44399232 IC50 = 21000000 nM T10965 CVDP57 44399253 IC50 > 50000000 nM T10965 C0ZIP8 44420653 IC50 = 2800 nM T10965 C5QXG3 44420654 IC50 = 3400 nM T10965 C2S9CH 44420657 IC50 = 1200 nM T10965 C8Y1HG 44420659 IC50 = 1100 nM T10965 CQ08EK 44420661 IC50 = 740 nM T10965 CA9T5O 44420662 IC50 = 3600 nM T10965 CCW67H 44566653 IC50 = 1000 nM T10965 CW8KR3 46845959 IC50 = 2500000 nM T10965 C8MUB4 46881482 IC50 = 11000000 nM T10965 CM2TE6 46881483 IC50 = 6500000 nM T10965 CE7OJ4 46881484 IC50 = 3000000 nM T10965 CS68ZT 46881485 IC50 = 5000000 nM T10965 COJ35S 46881517 IC50 = 11000000 nM T10965 CH0B8N 70789756 IC50 = 17000 nM T10965 CS1FC2 71450419 IC50 = 880000 nM T10965 CR8AC6 71452242 IC50 = 18000 nM T10965 CEPH60 71452644 IC50 = 22000 nM T10965 C0LI3S 71457566 IC50 > 1000000 nM T10965 CN0ZI6 71458017 IC50 = 7000 nM T10965 CF3TP8 71462945 IC50 > 1000000 nM T10965 C1NPL0 71552941 IC50 = 3100 nM T10965 CA4PS8 71552942 IC50 = 7400 nM T10965 CU2EL6 71553007 IC50 = 10000 nM T10965 C0EC4Z 71553008 IC50 = 6600 nM T10965 CK6CP5 71553010 IC50 = 7100 nM T10965 C3UA9C 71553011 IC50 = 1500 nM T10965 CEZ15Y 71553012 IC50 = 1200 nM T10965 CF1LY3 71553083 IC50 > 80000 nM T10965 C1CM5E 71553084 IC50 = 1100 nM T10965 CVIA91 71553085 IC50 = 400 nM T10965 CQ91EB 71553086 IC50 = 1200 nM T10965 CZM0S4 71553087 IC50 = 430 nM T10965 CJCE72 71553151 IC50 = 580 nM T10965 C1TR3O 71553152 IC50 = 2200 nM T10965 CH08XN 71553153 IC50 = 1600 nM T10965 CEN63Z 71553155 IC50 = 3000 nM T10965 CQZ8D4 71553156 IC50 > 80000 nM T10965 C5YN8K 71553236 IC50 = 3900 nM T10965 CGE8R2 71715994 IC50 = 420 nM T10965 C0FR3U 71716010 IC50 = 450 nM T10965 C3S7VA 71716029 IC50 = 1000000 nM T10965 C3JQ6N 71716030 IC50 = 70000 nM T10965 CEO6H7 71716031 IC50 = 540000 nM T10965 C6C0ZR 71716033 IC50 = 2000000 nM T10965 CJ2Q9U 71716626 IC50 = 1000000 nM T10965 C9R3XL 71717218 IC50 = 2 nM T10965 CS7T0Y 71717230 IC50 = 500000 nM T10965 C8V9FD 71717231 IC50 = 2000000 nM T10965 CK27AE 71717234 IC50 = 2000000 nM T10965 C8P0KB 71717843 IC50 = 2600000 nM T10965 CLN8X2 71717844 IC50 = 225000 nM T10965 CYT24W 71717846 IC50 = 17000000 nM T10965 C7NA8Z 71717847 IC50 = 12000000 nM T10965 CD31EA 71717849 IC50 = 2000000 nM T10965 CL25WA 71718488 IC50 = 20000000 nM T10965 CCO93Y 71719057 IC50 = 250000 nM T10965 CH42FQ 71719059 IC50 = 1000000 nM T10965 CBLP16 71719067 IC50 = 4900000 nM T10965 C8MHG7 71719069 IC50 = 12400000 nM T10965 CQR6H7 71719671 IC50 = 400000 nM T10965 C2XBN3 71719672 IC50 = 300000 nM T10965 CSMU14 71720272 IC50 = 2500000 nM T10965 C3Y5QT 71720273 IC50 = 200000 nM T10965 C7XR6V 71720274 IC50 = 700000 nM T10965 CTHW87 71720284 IC50 = 6900000 nM T10965 CCNR81 71720285 IC50 = 20000000 nM T10965 C3FIJ8 73354415 IC50 > 5000000 nM T10965 C8TE5P 76335199 IC50 = 100000 nM T10965 CJ9OU3 90664008 IC50 = 100 nM T10965 C0R2EU 90664042 IC50 = 60000 nM T10965 CB6QI0 90664073 IC50 = 1300 nM T10965 C52HET 90664075 IC50 = 900 nM T10965 CXH6L1 90664077 IC50 = 4300 nM T10965 CU0SM3 90664079 IC50 = 400 nM T10965 CU1LZ0 90664081 IC50 = 12000 nM T10965 CC9K8W 90664083 IC50 = 2400 nM T10965 C3YOJ9 90664085 IC50 = 1200 nM T10965 C1W2MK 90664087 IC50 = 100 nM T10965 C3QU9V 90664089 IC50 = 100 nM T10965 CJ4QK0 90664091 IC50 = 100 nM T10965 C8TWX7 90664093 IC50 = 600 nM T10965 C20WQE 90664095 IC50 = 12500 nM T10965 C80DNS 90664097 IC50 = 1700 nM T10965 C6D3UT 90664099 IC50 = 2500 nM T10965 CO2DA9 90664124 IC50 > 1000000 nM T10965 CKZP37 90664125 IC50 = 300000 nM T10965 CXN0Q3 90664160 IC50 = 380000 nM T10965 C86TFW 90664161 IC50 = 900000 nM T10965 C7V9EN 90664162 IC50 = 600000 nM T10965 C5ZKM2 90664163 IC50 = 26000 nM T10965 C2J7FQ 90664165 IC50 = 2000000 nM T10965 C49RXN 90664166 IC50 = 1500000 nM T10965 CUWF73 90664170 IC50 = 700000 nM T10965 CE1DY2 90664171 IC50 = 1000000 nM T10965 C13WQJ 90664172 IC50 = 160000 nM T10965 CDVW23 90664222 IC50 = 12000000 nM T10965 CJ3O0E 90664264 IC50 = 450 nM T10965 C6KN7R 90664265 IC50 = 2570 nM T10965 CF9XM7 118714544 IC50 = 520000 nM T10965 CZU9S3 118714545 IC50 = 18000 nM T10965 C6G1LI 118714546 IC50 = 34000 nM T10965 CIF1K3 118714547 IC50 = 8000 nM T10965 C9N2RD 118714548 IC50 = 19000 nM T10965 CI7C1S 118714549 IC50 = 21000 nM T10965 CX8D3J 118714550 IC50 = 16000 nM T10965 C6GY9S 118714551 IC50 = 8000 nM T10965 C15YGB 118719302 IC50 = 600 nM T10965 CI3VJ0 118719304 IC50 = 300 nM T10965 CZH6T3 118719305 IC50 = 300 nM T10965 C4BGF1 118719306 IC50 = 300 nM T10965 C2FX6G 135506443 IC50 = 130 nM T10965 C4BQ5L 135536082 IC50 = 290000 nM T10965 D00YPH 10239 IC50 = 6500000 nM T10965 D0E9NT 11874 IC50 = 11800 nM T10965 D0O6OH 71553154 IC50 = 1000 nM T10965 D0Y3TZ 370 IC50 = 19100 nM T07394 D09BXO 11261800 IC50 = 400 nM T07394 C2BGW0 16142 IC50 = 800 nM T07394 C6YMK0 441844 IC50 = 300 nM T07394 CU94QM 441874 IC50 = 2400 nM T07394 C9N5SF 2848109 IC50 = 4150 nM T07394 C5V6TP 3103157 IC50 = 2510 nM T07394 C8CZY4 11410873 IC50 = 300 nM T07394 CRZ49K 44387915 IC50 = 2000 nM T07394 C5PQ4Z 46210444 IC50 = 17300 nM T07394 CW68DS 71542548 IC50 = 2 nM T07394 C4Z9NE 71712019 IC50 = 4 nM T07394 C9W2QU 73441909 IC50 = 2 nM T07394 C37AFR 73441957 IC50 = 3 nM T07394 CLO08N 118732177 IC50 = 3 nM T07394 CLJ5Q3 118732178 IC50 = 1 nM T07394 CBUT48 118732179 IC50 = 13 nM T07394 CTD5J0 118732180 IC50 = 1190 nM T07394 CE4PC8 118732181 IC50 = 231 nM T07394 C7VA3N 118732182 IC50 = 32 nM T07394 CD2U5R 118732183 IC50 = 169 nM T07394 CY1ES6 118732184 IC50 = 54 nM T07394 CE7MX2 118732185 IC50 = 3 nM T07394 C64ACS 118732186 IC50 = 1 nM T07394 C6MUQ2 118732187 IC50 = 3 nM T07394 CH4YL5 118732188 IC50 = 2060 nM T07394 CEGM19 118732189 IC50 = 9 nM T07394 C4WY7T 118732190 IC50 = 2 nM T07394 CKE83Y 118732191 IC50 = 1 nM T07394 CWC0U9 118732192 IC50 = 2 nM T07394 CZ19PD 145954977 IC50 = 700 nM T07394 C46LTO 145979138 IC50 = 3320 nM T07394 C1W8LD 145979748 IC50 = 330 nM T07394 C62MZI 145979931 IC50 > 10000 nM T07394 C9D6RC 145980768 IC50 > 10000 nM T07394 CZ73PS 145980911 IC50 = 4270 nM T07394 CR42PF 145980992 IC50 = 43200 nM T07394 CSB3W7 145981132 IC50 = 1520 nM T07394 C3DSG1 145982044 IC50 > 10000 nM T07394 C3GCL9 145982920 IC50 = 2950 nM T07394 C8A4DF 145987925 IC50 = 2590 nM T07394 CV2M1I 145988452 IC50 = 760 nM T07394 CNK94B 145988996 IC50 = 770 nM T07394 C3GPR4 145989833 IC50 = 860 nM T07394 C7GO0Y 145989905 IC50 > 10000 nM T07394 C8F6RV 145989989 IC50 > 10000 nM T07394 CW5OK3 145991181 IC50 = 220 nM T07394 CC30AX 145991872 IC50 = 360 nM T07394 C2SBN0 145992082 IC50 > 10000 nM T07394 C8U3MK 145992650 IC50 = 640 nM T07394 CVW02L 145992893 IC50 = 130 nM T07394 CS3BQ1 145993024 IC50 = 14700 nM T07394 CO6FC0 145993456 IC50 = 12300 nM T01597 CH0ZD7 207299 IC50 > 100000 nM T01597 CB27WS 849733 IC50 > 10000 nM T01597 CJ6RO8 122193596 IC50 > 10000 nM T01597 C46ISV 127038222 IC50 > 100000 nM T84581 CMYC68 271296 IC50 = 2400 nM T84581 CI2KV3 637858 IC50 = 45880 nM T84581 CHKN64 139035059 IC50 = 960 nM T84581 CAVG72 145979255 IC50 = 783 nM T84581 C9F6JU 155514175 IC50 > 200000 nM T84581 CUI8K4 155516107 IC50 > 200000 nM T84581 CX5R8U 155519730 IC50 > 200000 nM T84581 CVZH61 155521770 IC50 = 6610 nM T84581 CS80HU 155522405 IC50 = 5280 nM T84581 CUY7D0 155527965 IC50 = 81630 nM T84581 CX9E7P 155531650 IC50 = 30540 nM T84581 CV3A6Z 155539709 IC50 = 76620 nM T84581 C5WS1Z 155552949 IC50 = 29300 nM T84581 CZL2M5 155558702 IC50 = 820 nM T84581 CJVI42 155565055 IC50 = 16010 nM T84581 CS8D4G 155568338 IC50 = 2510 nM T84581 D04FNI 11657687 IC50 = 4600 nM T84581 D05CCT 4139 IC50 = 30000 nM T53251 D02HFD 124886 IC50 > 100000 nM T53251 D07BDD 65359 IC50 > 100000 nM T53251 D09FAZ 9444 IC50 > 10000 nM T53251 D0V0LB 6058 IC50 > 100000 nM T53251 D0X5SD 3117 IC50 = 600 nM T53251 D0X5XU 451668 IC50 > 10000 nM T53251 D0B1FE 3194 IC50 = 400 nM T53251 D09YFD 21928 IC50 = 1200 nM T53251 D0X2AU 23427 IC50 = 4400 nM T53251 D0N1XD 6223 IC50 = 530 nM T53251 CF3N7H 5941 IC50 = 15000 nM T53251 C8IWZ0 10236 IC50 = 54000 nM T53251 CGJ83B 15460 IC50 = 550 nM T53251 CX1LG8 65093 IC50 = 650 nM T53251 C95WZA 123446 IC50 = 790 nM T53251 CY2ON3 194564 IC50 > 100000 nM T53251 CJ7FR6 533728 IC50 = 9200 nM T53251 C37UOC 590397 IC50 = 450 nM T53251 CKH28J 1926147 IC50 = 39030 nM T53251 C91GWT 3007092 IC50 = 2100 nM T53251 CU54KV 3084126 IC50 = 630 nM T53251 CQE8T5 5462814 IC50 = 500 nM T53251 CO04SL 9883072 IC50 = 55000 nM T53251 CQS5Z1 10417379 IC50 = 170 nM T53251 CA5S0G 11667575 IC50 = 4897.79 nM T53251 CZV31A 13989137 IC50 = 2600 nM T53251 CGR64Y 13989139 IC50 = 58000 nM T53251 C8RD2F 15608594 IC50 = 10600 nM T53251 C6GNZ9 15608600 IC50 = 27100 nM T53251 CBX8T9 16451230 IC50 > 150000 nM T53251 C4IAR3 16645216 IC50 > 100000 nM T53251 CFR03M 20867934 IC50 = 6890 nM T53251 CK1Y7A 20867935 IC50 = 1220 nM T53251 C7ZNU6 20867937 IC50 = 5970 nM T53251 CB8M4Y 20867956 IC50 = 3750 nM T53251 CL32YO 20867958 IC50 = 2180 nM T53251 CPG38H 20867975 IC50 = 3470 nM T53251 C9ALV6 20867976 IC50 = 3870 nM T53251 C85NAQ 24858111 IC50 > 10000 nM T53251 C5N3LG 44251522 Ki = 2.6 nM T53251 CCI45D 44604812 IC50 = 9 nM T53251 CB1Z5L 44604813 IC50 > 10000 nM T53251 CQ0C4W 44604814 IC50 > 10000 nM T53251 CB53JP 44604815 IC50 = 3877 nM T53251 C8Z4RA 44604816 IC50 = 5100 nM T53251 CZS90V 44604817 IC50 = 5800000 nM T53251 CBIV83 44605024 IC50 = 200 nM T53251 CFU9H7 44605025 IC50 = 31 nM T53251 CL76QF 44605026 IC50 = 1600 nM T53251 CFQ17S 44605027 IC50 = 343 nM T53251 C6PY2V 44605028 IC50 = 191 nM T53251 CEY32T 44605029 IC50 = 9100 nM T53251 CFE1B9 44607518 IC50 > 1000 nM T53251 C4I9OP 46174171 IC50 = 123 nM T53251 CZF8V7 46174173 IC50 = 160 nM T53251 C7LT8D 46191942 IC50 = 1700 nM T53251 CE85SN 46192084 IC50 > 50000 nM T53251 CP98TY 46192085 IC50 > 50000 nM T53251 C6QZM4 46885506 IC50 > 10000 nM T53251 CXG8N1 46899643 IC50 = 910000 nM T53251 CO31AG 46899644 IC50 > 10000000 nM T53251 C5NQ4C 46901285 IC50 = 110000 nM T53251 CLM1Z5 46901453 IC50 = 110000 nM T53251 C2JC1D 46901454 IC50 = 49000 nM T53251 C0QES1 46901455 IC50 = 3200000 nM T53251 CR5O3X 46901456 IC50 = 41000 nM T53251 C17FAV 46901457 IC50 = 65000 nM T53251 CYL37W 46901621 IC50 = 51000 nM T53251 C9YA2R 46901622 IC50 = 8 nM T53251 CP5W2T 46901623 IC50 = 910 nM T53251 C3FX7W 46901624 IC50 = 780000 nM T53251 C0UQ4R 46901625 IC50 = 3400 nM T53251 C3WUF9 46901785 IC50 > 10000 nM T53251 C3SI5T 46901786 IC50 > 10000000 nM T53251 CQ46GJ 46901787 IC50 = 235000 nM T53251 C98UPC 46901788 IC50 > 10000000 nM T53251 CK6N7P 46901789 IC50 = 57000 nM T53251 C62KOY 46901935 IC50 = 173000 nM T53251 CO7IF4 46901936 IC50 = 1500000 nM T53251 CK56RG 46902073 IC50 > 10000000 nM T53251 C1EQK6 46902074 IC50 > 10000000 nM T53251 CM8Z1G 53303486 IC50 = 26400 nM T53251 CDW86Q 53315436 IC50 = 101 nM T53251 C6DUZ5 53315437 IC50 = 472 nM T53251 CT05PV 53315811 IC50 = 10 nM T53251 C2SY4X 53315855 IC50 = 8 nM T53251 C6SFC5 53315860 IC50 = 31 nM T53251 C18FDR 53315861 IC50 = 2 nM T53251 CKQ4R9 53315862 IC50 = 100 nM T53251 C9VAH6 53315863 IC50 = 7 nM T53251 C2HEM1 53315864 IC50 < 2.5 nM T53251 CAXE92 53315865 IC50 = 470 nM T53251 C3A5PI 53315866 IC50 < 2.5 nM T53251 CGMK45 53315867 IC50 = 9 nM T53251 CBE2L9 53315868 IC50 = 4 nM T53251 CPOX26 53315874 IC50 = 180 nM T53251 C8LR4J 53315875 IC50 = 260 nM T53251 CA8BC6 53315877 IC50 = 10 nM T53251 C7V6OX 53315879 IC50 = 56 nM T53251 C70VHB 53315882 IC50 = 6 nM T53251 C02ORV 53377508 Ki > 20000 nM T53251 CG0QW1 53921867 IC50 = 14400 nM T53251 CPL71I 54596764 IC50 > 100000 nM T53251 C72GHW 56642706 IC50 > 100000 nM T53251 CS6Q7R 56642708 IC50 > 100000 nM T53251 CV8A4S 56676725 IC50 = 106 nM T53251 C01NZY 57333568 IC50 > 100000 nM T53251 CER5F1 67466175 IC50 > 100000 nM T53251 C5QE6A 67988955 IC50 > 50000 nM T53251 CAVD69 70678415 IC50 = 20000 nM T53251 CGZ5P0 71521184 IC50 = 13100 nM T53251 CEP06B 71566707 IC50 = 5200 nM T53251 CV58PD 71716146 IC50 = 3300 nM T53251 C1GUK2 71716147 IC50 = 23500 nM T53251 C07EOT 71717376 IC50 > 100000 nM T53251 CA7LC2 71718585 IC50 = 5300 nM T53251 CDX7M1 71718586 IC50 = 7200 nM T53251 CSTZ09 71730327 IC50 = 3190 nM T53251 CNU5Q1 71738181 IC50 = 1326 nM T53251 CK3P0Z 71738259 IC50 = 576 nM T53251 CN2HU1 71738262 IC50 = 506 nM T53251 CF58AV 71738398 IC50 = 10000 nM T53251 C1HZ4K 71738399 IC50 > 10000 nM T53251 CCZ57A 71738401 IC50 > 10000 nM T53251 CXJ14A 71738402 IC50 = 1000 nM T53251 CDI3K7 71738471 IC50 = 344 nM T53251 CNRD47 71738474 IC50 > 1000 nM T53251 CR8M7D 71738544 IC50 = 10000 nM T53251 CUJ2O0 71738546 IC50 > 10000 nM T53251 C98AFK 71738604 IC50 > 10000 nM T53251 CVC94H 71738605 IC50 = 1000 nM T53251 CUT4Z1 71738606 IC50 = 830 nM T53251 C8Y5OC 71738608 IC50 > 10000 nM T53251 CG54BU 71738681 IC50 > 1000 nM T53251 CKN03R 71738741 IC50 > 10000 nM T53251 CK7OL8 72714452 IC50 < 2.5 nM T53251 C2PGX6 72714453 IC50 = 14 nM T53251 C67RUI 72714542 IC50 = 26 nM T53251 CS9HG2 72714543 IC50 = 310 nM T53251 C1ET0H 72714544 IC50 = 4 nM T53251 C5S8TC 72714643 IC50 > 26000 nM T53251 CM0WF1 72714644 IC50 > 50000 nM T53251 C5Q3OK 72714730 IC50 = 9 nM T53251 CF56EA 76310296 IC50 = 18200 nM T53251 CSTO69 76310297 IC50 = 5 nM T53251 CU7YP6 76310298 IC50 = 3.7 nM T53251 CZI95J 76313973 IC50 = 18 nM T53251 CT6S7V 76317517 IC50 = 4.8 nM T53251 CZ38OQ 76317518 IC50 = 0.9 nM T53251 C2K6JB 76324862 IC50 = 1342 nM T53251 C3INO2 76328419 IC50 = 2460 nM T53251 C7O4AC 76328420 IC50 = 3540 nM T53251 C5LQP0 76328421 IC50 = 754 nM T53251 CNLQ10 76332100 IC50 = 1 nM T53251 CK9YO4 76332101 IC50 = 12900 nM T53251 CWZC50 76335720 IC50 = 153 nM T53251 C2Q3SE 76335721 IC50 = 150 nM T53251 C4XJ5N 78357767 IC50 > 100000 nM T53251 CCT09O 86288827 IC50 = 103000 nM T53251 C01DAP 86288828 IC50 = 1600 nM T53251 CHDI72 89821586 IC50 > 50000 nM T53251 C6NA3U 90063226 IC50 < 3 nM T53251 CA18TS 90655765 IC50 = 190000 nM T53251 C5NX4U 90655766 IC50 = 157000 nM T53251 C18ICL 101882806 IC50 = 13 nM T53251 C8Z2HS 101882807 IC50 = 21 nM T53251 CGI15N 117915100 IC50 = 690 nM T53251 CB01GN 117915102 IC50 = 78 nM T53251 CPI53S 118607332 IC50 = 30 nM T53251 CSTY10 118607373 IC50 = 838 nM T53251 C9BI8F 118607414 IC50 = 0.5 nM T53251 CSW92P 118607432 IC50 = 8 nM T53251 CO1D7I 118607435 IC50 = 17 nM T53251 C6PZ1X 118607459 IC50 = 2060 nM T53251 CBA79J 118607465 IC50 = 859 nM T53251 CLS25W 118607471 IC50 = 6 nM T53251 C1K0VJ 118607474 IC50 = 27 nM T53251 C8XMV5 118607488 IC50 = 2 nM T53251 CY1X2K 118613614 IC50 = 532 nM T53251 CT6OD8 118613615 IC50 = 3140 nM T53251 COPW27 118613616 IC50 = 1080 nM T53251 CJW05H 118613617 IC50 = 7 nM T53251 C7X2AQ 118613624 IC50 = 22 nM T53251 CE69HN 118613626 IC50 = 146 nM T53251 CDK3F2 118613628 IC50 = 105 nM T53251 C5AF9V 118613631 IC50 = 2720 nM T53251 CG39ZR 118613632 IC50 = 52 nM T53251 CUDE80 118613633 IC50 = 44 nM T53251 CLIZ07 118613634 IC50 = 43 nM T53251 CG6E0J 118613636 IC50 = 15 nM T53251 C07LSQ 118613637 IC50 = 40 nM T53251 CB0K3S 118613639 IC50 = 0.5 nM T53251 C7SIL0 118613641 IC50 = 142 nM T53251 CQD69N 118613646 IC50 = 2 nM T53251 CQNA84 118613647 IC50 = 11 nM T53251 CBC0Q9 118613651 IC50 = 76 nM T53251 C2EQ9X 118613653 IC50 = 15 nM T53251 C1X8GW 118613658 IC50 = 63 nM T53251 C0JVC9 118613660 IC50 = 12 nM T53251 CI70WP 118613691 IC50 = 94 nM T53251 CQ5T3E 118613693 IC50 = 637 nM T53251 CFGK68 118613694 IC50 = 48 nM T53251 C1LOF4 118613696 IC50 = 15 nM T53251 CAY5Q6 118613697 IC50 = 264 nM T53251 CG7D9I 118613701 IC50 = 42 nM T53251 C3ZJO5 118613702 IC50 = 136 nM T53251 COJB60 118613705 IC50 = 6 nM T53251 CX8J7D 118613718 IC50 = 148 nM T53251 CKI70Y 118613722 IC50 = 699 nM T53251 CJY8E1 118613723 IC50 = 244 nM T53251 CPW12K 118613724 IC50 = 436 nM T53251 C3QX6D 118613726 IC50 = 6 nM T53251 CKO15P 118613728 IC50 = 735 nM T53251 CW1D6K 118613729 IC50 = 16 nM T53251 CV0FW8 121225442 IC50 = 99000 nM T53251 C6G0CZ 122580323 EC50 > 100000 nM T53251 C7TI9A 129012136 IC50 = 295 nM T53251 C6F2VK 129012137 IC50 = 259 nM T53251 CJI14M 129072680 IC50 = 351 nM T53251 CU3FP1 129072681 IC50 = 1150 nM T53251 C0ES4L 129072695 IC50 = 1450 nM T53251 COL81P 129085358 IC50 = 18 nM T53251 CUZ6K0 129085359 IC50 = 6110 nM T53251 CI1H4A 129085361 IC50 = 342 nM T53251 C2B5VP 129085364 IC50 = 24 nM T53251 CJ18GA 129085365 IC50 = 21 nM T53251 CUO5E6 129085366 IC50 = 123 nM T53251 CVPH43 129085367 IC50 = 599 nM T53251 CKS08I 129085368 IC50 = 3910 nM T53251 CNO1K2 129085369 IC50 = 7550 nM T53251 CIST32 129085377 IC50 = 3080 nM T53251 CL9KB8 129246684 IC50 = 2870 nM T53251 C6ZYB8 129270457 IC50 = 935 nM T53251 CTQE45 132471834 IC50 = 318 nM T53251 CBO31X 132471835 IC50 = 177 nM T53251 CL2ZI0 132609264 IC50 = 67200 nM T53251 CYJR92 132609265 IC50 = 39600 nM T53251 CC9T8K 134133015 IC50 = 3960 nM T53251 CT6OU2 134135896 IC50 = 4570 nM T53251 C1AHT2 134136303 IC50 = 4840 nM T53251 CIF53U 134140514 IC50 = 3840 nM T53251 CQ5G7S 134141610 IC50 = 2490 nM T53251 CK6WC2 134142720 IC50 = 2980 nM T53251 C9C4XA 134144529 IC50 = 2680 nM T53251 CY8EG2 134145804 IC50 = 3480 nM T53251 CF9P7V 134146800 IC50 = 1870 nM T53251 CX34OF 134149718 IC50 = 3220 nM T53251 C0AOE3 134397507 IC50 = 6 nM T53251 C6GC0O 137028680 EC50 > 100000 nM T53251 C4S1ZI 137333995 Ki = 3.6 nM T53251 CBTH20 137348638 IC50 = 992 nM T53251 C5ZM8O 137628302 IC50 > 100000 nM T53251 CR53YC 137631913 IC50 = 92 nM T53251 C8VO5D 137632076 IC50 = 756 nM T53251 C5AC6M 137632524 IC50 = 532 nM T53251 C46WLE 137633319 IC50 > 6000 nM T53251 CIB30Q 137633627 IC50 = 438 nM T53251 C8AM9L 137635489 IC50 = 4070 nM T53251 CE60DR 137635748 IC50 = 313 nM T53251 CTU4G0 137636690 IC50 = 481 nM T53251 CI5Q3X 137636915 IC50 = 323 nM T53251 CK1WU6 137637870 IC50 = 359 nM T53251 C3TD2E 137638286 IC50 = 262 nM T53251 CO6JA8 137639333 IC50 > 5000 nM T53251 CO78IY 137639766 IC50 = 484 nM T53251 C0EYN9 137639969 IC50 = 282 nM T53251 CCSI40 137640754 IC50 = 356 nM T53251 C2P3JR 137640823 IC50 = 169000 nM T53251 C5TY4L 137640829 IC50 = 1160 nM T53251 C7G9AB 137643064 IC50 = 534 nM T53251 CV4PI3 137643498 IC50 > 6000 nM T53251 C2DWX9 137643972 IC50 = 191300 nM T53251 CZM39K 137644029 IC50 = 3690 nM T53251 CS9RO5 137644870 IC50 = 110 nM T53251 C6NW5B 137645215 IC50 = 788 nM T53251 C6WLD1 137645686 IC50 = 224 nM T53251 CZTV84 137646234 IC50 = 311 nM T53251 C9EP0L 137647456 IC50 = 1630 nM T53251 CN5UY2 137647689 IC50 > 5000 nM T53251 CD2JQ9 137648196 IC50 = 956 nM T53251 CJO19V 137649514 IC50 = 1582 nM T53251 CZD47A 137649599 IC50 = 436 nM T53251 CZR86C 137650174 IC50 = 151 nM T53251 CSU4J8 137651295 IC50 = 1060 nM T53251 CJ57XR 137652778 IC50 = 1150 nM T53251 C8N2BU 137653025 IC50 = 313 nM T53251 C4JYZ0 137654123 IC50 = 1910 nM T53251 CES2Y4 137654330 IC50 = 726 nM T53251 CF65YG 137654447 IC50 = 465 nM T53251 CX2RM3 137654889 IC50 = 724 nM T53251 C8MQ2I 137655652 IC50 = 585 nM T53251 C3BI4K 137655660 IC50 = 407 nM T53251 CHS71L 137656981 IC50 = 508 nM T53251 CYF6V9 137657228 IC50 = 315 nM T53251 C0R6QN 137658284 IC50 = 341 nM T53251 CR7GF2 137658708 IC50 = 190 nM T53251 CDQW60 137661215 IC50 > 5000 nM T53251 C19VQE 137661488 IC50 = 443 nM T53251 CD1K7J 137661663 IC50 = 306 nM T53251 C85XIG 137662224 IC50 = 550 nM T53251 C8LEV4 139267760 IC50 > 10000 nM T53251 CEUV89 139592901 IC50 = 6438 nM T53251 C4QV0A 145433713 IC50 = 27370 nM T53251 C95RGF 145950703 IC50 = 3 nM T53251 C0XBU5 145951018 IC50 = 3 nM T53251 CIKY95 145954902 IC50 = 336 nM T53251 C5NS1C 145963999 IC50 = 3220 nM T53251 CMX3R9 145964677 IC50 = 115 nM T53251 C7XF6P 145965645 IC50 = 5410 nM T53251 CW2ZV7 145967174 IC50 = 5 nM T53251 C39OCT 145967367 IC50 = 3260 nM T53251 C3JO8Q 145971403 IC50 = 5130 nM T53251 COJG25 145974212 IC50 = 21 nM T53251 CKVI47 145974419 IC50 = 378 nM T53251 CW1LX9 145975217 IC50 = 41 nM T53251 CIP42V 145976082 IC50 = 7 nM T53251 C8MFK6 145977537 IC50 = 13 nM T53251 C5I0ZL 145977690 IC50 = 1470 nM T53251 CU2A1M 145978072 IC50 = 13 nM T53251 C3MF6X 145978745 IC50 = 3450 nM T53251 CZXL32 145979245 IC50 = 295 nM T53251 C7J5EC 145979293 IC50 = 332 nM T53251 C3RU0V 145979319 IC50 = 46830 nM T53251 CPOD29 145979530 IC50 = 55 nM T53251 CT5J4M 145980087 IC50 = 575 nM T53251 CP45HE 145980274 IC50 = 869 nM T53251 CR21UC 145980408 IC50 = 114 nM T53251 CCZ04N 145980685 IC50 = 2034 nM T53251 C95KTO 145981287 IC50 = 319 nM T53251 CBN7A4 145982061 IC50 = 55 nM T53251 CO37UP 145982259 IC50 = 132 nM T53251 CZA3O1 145982342 IC50 = 119 nM T53251 C8SQU6 145982395 IC50 > 50000 nM T53251 C7T4AF 145986487 IC50 = 211 nM T53251 CU09KV 145986544 IC50 = 223 nM T53251 CUIM15 145986653 IC50 = 8 nM T53251 CC0T5D 145986874 IC50 = 46970 nM T53251 C3P9ZS 145987918 IC50 = 116 nM T53251 CL7QM9 145988523 IC50 = 39 nM T53251 CRNQ80 145988862 IC50 = 116 nM T53251 C2GVW8 145988903 IC50 = 10000 nM T53251 C0HE8L 145988989 IC50 = 169 nM T53251 CD0V1H 145989374 IC50 > 25000 nM T53251 C2JU8Y 145989377 IC50 = 185 nM T53251 C3L6QS 145989766 IC50 = 843 nM T53251 C3RVN1 145989815 IC50 = 1018 nM T53251 CB7AH5 145990230 IC50 = 128 nM T53251 CLJS40 145990269 IC50 = 4 nM T53251 C9SY1K 145990579 IC50 = 123 nM T53251 C0BND7 145990594 IC50 = 112 nM T53251 C84GQH 145990877 IC50 = 25 nM T53251 CZH9D6 145990892 IC50 = 683 nM T53251 CB7J2S 145990975 IC50 = 5344 nM T53251 CR2Q5I 145991323 IC50 = 37790 nM T53251 CWYX53 145991364 IC50 = 1214 nM T53251 C1SKL0 145991772 IC50 = 49 nM T53251 CR84CL 145991918 IC50 = 39 nM T53251 C2H0LX 145993122 IC50 = 1000 nM T53251 CFC96O 145993541 IC50 > 1000 nM T53251 C7MHP1 145993725 IC50 = 1000 nM T53251 CJ64RU 145993764 IC50 = 10 nM T53251 C2ST6R 145993977 IC50 = 7136 nM T53251 C3HY6V 145994014 IC50 = 1000 nM T53251 CJT6G1 155511077 IC50 = 358 nM T53251 CRV06Z 155511081 IC50 = 30100 nM T53251 C4NS2X 155512777 IC50 = 20100 nM T53251 CO5P4T 155513225 IC50 = 142 nM T53251 CW0C4P 155517779 IC50 > 100000 nM T53251 CB9WP0 155517958 IC50 = 1350 nM T53251 CFLK08 155520544 IC50 = 648 nM T53251 CYOD10 155522526 IC50 = 3580 nM T53251 CJOW75 155522891 IC50 = 32 nM T53251 CL4T2Q 155523641 IC50 = 1900 nM T53251 C4UXQ1 155526805 IC50 = 1220 nM T53251 CLQ18S 155527069 IC50 = 2340 nM T53251 CP60DZ 155527429 IC50 = 3280 nM T53251 CG2EM1 155527465 IC50 = 81300 nM T53251 CH5X4E 155527661 IC50 = 219 nM T53251 CD8C5B 155528012 IC50 = 1200 nM T53251 CKN4C6 155528155 IC50 = 15 nM T53251 CX5G9E 155528619 EC50 = 31800 nM T53251 C53YIH 155530887 IC50 = 30 nM T53251 C94QSB 155531144 IC50 = 120 nM T53251 CA9P6Y 155532307 IC50 = 21 nM T53251 C1J5TI 155532811 IC50 = 2450 nM T53251 CAE51Q 155534378 EC50 = 50900 nM T53251 CI0ML6 155534407 IC50 = 3640 nM T53251 C7YKH1 155535402 IC50 = 3100 nM T53251 C6FEP9 155535898 IC50 = 3020 nM T53251 CU2XG3 155537180 IC50 = 4780 nM T53251 C7Q9HD 155537279 IC50 = 107 nM T53251 C6R7JS 155537616 IC50 = 211 nM T53251 C78EAT 155538085 IC50 = 447 nM T53251 C5OGN0 155542626 IC50 = 1630 nM T53251 CHL9F7 155543202 IC50 = 18900 nM T53251 C0VJO4 155545582 IC50 = 19100 nM T53251 CBLI45 155547053 IC50 = 2540 nM T53251 C51VKD 155547438 IC50 = 61 nM T53251 CQ4X5G 155549294 IC50 = 2984 nM T53251 C8Q3GX 155550036 IC50 = 1190 nM T53251 CMLA31 155550222 IC50 = 955 nM T53251 CSKE02 155550699 IC50 = 9230 nM T53251 C1QOP9 155550708 IC50 = 47 nM T53251 CJO5H8 155553691 IC50 = 1090 nM T53251 CTIM98 155556005 IC50 = 338 nM T53251 CIN57Q 155556138 EC50 = 142400 nM T53251 CZQP24 155556616 IC50 = 900 nM T53251 CVT50L 155557402 IC50 = 740 nM T53251 CB8SD4 155557649 EC50 = 137000 nM T53251 CYAP13 155557747 IC50 = 163 nM T53251 C5KZP1 155558337 IC50 = 214 nM T53251 CQ08KG 155559900 IC50 = 4540 nM T53251 C2FIO6 155559947 IC50 = 6840 nM T53251 CM94DV 155560212 IC50 = 10000 nM T53251 CW92RC 155560401 IC50 = 2091 nM T53251 CD3HO4 155562561 IC50 = 7960 nM T53251 C0J6AT 155562781 IC50 = 359 nM T53251 C5VN8K 155564441 IC50 = 6170 nM T53251 CVZ2C4 155565339 IC50 = 672 nM T53251 C84AKC 155566143 IC50 = 14 nM T53251 D00FLT 65482 IC50 = 509000 nM T53251 D02TVQ 71268957 IC50 > 100000 nM T53251 D02UVS 5455 IC50 = 550 nM T53251 D04FNI 11657687 IC50 = 2400 nM T53251 D06PPL 25150857 IC50 = 67 nM T53251 D09CLP 439155 Ki = 570 nM T53251 D0BI4T 53315878 IC50 < 2.5 nM T53251 D0C5EG 76285486 IC50 = 3 nM T53251 D0CX4W 46901937 IC50 = 9000 nM T53251 D0DQ6Z 8530 IC50 = 2000 nM T53251 D0GK7A 46224516 Ki = 3.7 nM T53251 D0L5LN 6780 IC50 > 100000 nM T53251 D0LA0P 72193870 EC50 = 5000 nM T53251 D0RO9T 73755260 IC50 = 1500 nM T96413 C0X4MN 122306 IC50 = 45750 nM T96413 COLK49 404566 IC50 = 456600 nM T96413 CVR7D9 101879515 IC50 = 900 nM T96413 CZ7E8Q 122180089 IC50 = 46140 nM T96413 CX3RK4 122180090 IC50 = 8140 nM T96413 C3WZ9E 122180091 IC50 = 11140 nM T96413 C9C2TD 122180092 IC50 = 15140 nM T96413 CUKF85 122180093 IC50 = 19160 nM T96413 CP57WK 122180095 IC50 = 13140 nM T96413 C2V5YM 122180096 IC50 = 4120 nM T96413 C5AF4E 122180097 IC50 = 16120 nM T96413 CH12ZP 122180100 IC50 = 30140 nM T96413 CER37M 122180101 IC50 = 32140 nM T96413 C0NX3R 122180102 IC50 = 40140 nM T96413 C9ET3G 122180103 IC50 = 31140 nM T96413 CK1IH2 122180106 IC50 = 20140 nM T96413 CPF4D6 127048343 IC50 = 18000 nM T96413 CF4UN1 127048344 IC50 = 22300 nM T96413 CWZ95L 127048345 IC50 = 38500 nM T96413 C3SLV1 127048693 IC50 = 51000 nM T96413 CTE49Y 127048694 IC50 = 80100 nM T96413 CIO20X 127048695 IC50 = 69400 nM T96413 CXLW15 127049986 IC50 = 16600 nM T96413 C5T3UC 127049987 IC50 = 78900 nM T96413 C15AGJ 127049988 IC50 = 44100 nM T96413 CI0C4R 127049989 IC50 = 19400 nM T96413 CH5XS7 127049990 IC50 = 68380 nM T96413 C8U5JT 127049991 IC50 = 49380 nM T96413 CQEV18 127050225 IC50 = 42250 nM T96413 C9R8NQ 127051486 IC50 = 38500 nM T96413 CVAJ82 127051487 IC50 = 18100 nM T96413 C59EFN 127051489 IC50 = 46140 nM T96413 CGOV82 127052074 IC50 = 26300 nM T96413 C94OTL 127052404 IC50 = 9200 nM T96413 C7S8LM 127052440 IC50 = 46100 nM T96413 CN0E6T 127053019 IC50 = 18400 nM T96413 CRZ1B9 127053020 IC50 = 24200 nM T96413 CED51R 127053021 IC50 = 37010 nM T96413 CD1R6Q 135400456 IC50 = 177000 nM T96413 C9PI7O 135402338 IC50 = 20100 nM T96413 C0HQF2 135404247 IC50 = 39800 nM T96413 C95RAN 135405744 IC50 = 22200 nM T96413 CG8D0A 135412164 IC50 = 1800 nM T96413 CM5Q1Z 135430309 IC50 = 1100 nM T96413 C9G3NT 135436839 IC50 = 61030 nM T96413 CA0R7X 135452109 IC50 = 172700 nM T96413 CEM0L4 135458774 IC50 = 10000 nM T96413 CR80IZ 135460530 IC50 = 5500 nM T96413 CYS5U3 135470028 IC50 = 120500 nM T96413 CXR4A9 135484663 IC50 = 600 nM T96413 C14KRW 135501581 IC50 = 2100 nM T96413 CBK98Y 135502629 IC50 = 50400 nM T96413 C09XWB 135503134 IC50 = 1500 nM T96413 CR56ZO 135567246 IC50 = 198200 nM T96413 C0IZD8 135567247 IC50 = 2100 nM T96413 CX70BW 135995892 IC50 = 3140 nM T96413 CF8VK5 135995893 IC50 = 2140 nM T96413 CXY9I2 136006573 IC50 = 700 nM T96413 C4HJ7D 136044076 IC50 = 2800 nM T96413 C46VDR 136044077 IC50 = 37700 nM T96413 CNPL62 136044078 IC50 = 1170 nM T96413 C8A1SE 136044079 IC50 = 3200 nM T96413 CV01GC 136044080 IC50 = 30900 nM T96413 C79OIG 136044081 IC50 = 1800 nM T96413 CBF97D 136044082 IC50 = 44000 nM T96413 CKTI80 136094794 IC50 = 9600 nM T96413 CM5SQ1 136094795 IC50 = 6700 nM T96413 CYS27J 136998773 IC50 = 29250 nM T96413 C9GIY5 136998774 IC50 = 46100 nM T96413 C04UBX 137224958 IC50 = 9600 nM T96413 CSQU45 137224959 IC50 = 8300 nM T96413 CD1T8O 137225017 IC50 = 5010 nM T96413 C1OQ5Y 137225018 IC50 = 2600 nM T96413 CPW6R7 137225049 IC50 = 3100 nM T96413 CHN2Y6 137225050 IC50 = 2110 nM T96413 CX9E3A 145949237 IC50 = 1100 nM T96413 CH7DQ3 145949733 IC50 = 300 nM T96413 CM9C3G 145950464 IC50 = 33500 nM T96413 CA60NG 145950743 IC50 = 2980 nM T96413 C7FCH6 145950828 IC50 = 23400 nM T96413 CEU95S 145951044 IC50 = 2800 nM T96413 CNPO25 145951171 IC50 = 300 nM T96413 CB3UX2 145951999 IC50 = 42750 nM T96413 C87THG 145952382 IC50 = 2200 nM T96413 C67XIQ 145953043 IC50 = 3448 nM T96413 CG0TK9 145953889 IC50 = 100 nM T96413 CEPV32 145954312 IC50 = 2670 nM T96413 CBI8V7 145954569 IC50 = 1200 nM T96413 C2Z5DG 145955659 IC50 = 100 nM T96413 C0O3XW 145956092 IC50 = 43500 nM T96413 CJ35ZM 145957178 IC50 = 5874 nM T96413 C13QPB 145957270 IC50 = 48500 nM T96413 CIZ18M 145957921 IC50 = 22200 nM T96413 C2ZS4K 145958298 IC50 = 5800 nM T96413 CDV73H 145958392 IC50 = 13100 nM T96413 CI7EF0 145958395 IC50 = 12500 nM T96413 CFI47P 145959449 IC50 = 7571 nM T96413 CAVT57 145959898 IC50 = 1140 nM T96413 CFA4L2 145959952 IC50 = 2100 nM T96413 C63WYX 145960254 IC50 = 32900 nM T96413 C85CEI 145960255 IC50 = 6900 nM T96413 CFDU52 145960276 IC50 = 32800 nM T96413 CJ07YB 145961856 IC50 = 15800 nM T96413 C30QZN 145962484 IC50 = 2348 nM T96413 CWL4A6 145971217 IC50 = 1500 nM T96413 CB9A3J 145971995 IC50 = 200 nM T96413 CEU05W 145972650 IC50 = 2800 nM T96413 C8O6CR 155518480 IC50 = 34160 nM T96413 CAVH63 155523289 IC50 = 5140 nM T96413 CSLQ70 155524682 IC50 = 12300 nM T96413 CW7LS9 155528641 IC50 = 7600 nM T96413 CL2VW7 155528982 IC50 = 1400 nM T96413 C5ZQT3 155530517 IC50 = 26140 nM T96413 C8T0UZ 155532176 IC50 = 56100 nM T96413 CG7U0L 155543919 IC50 = 27600 nM T96413 CCW5G4 155547952 IC50 = 46460 nM T96413 CP2SQ3 155554484 IC50 = 58160 nM T96413 CLU9V2 155555883 IC50 = 17200 nM T96413 C5SH7F 155558105 IC50 = 2600 nM T96413 CV6O4Y 155558317 IC50 = 960 nM T96413 C0Q3DY 155560145 IC50 = 6200 nM T96413 CH6N3F 155562800 IC50 = 28100 nM T96413 C61SOJ 155562831 IC50 = 8200 nM T96413 C2Y9WU 155565514 IC50 = 15300 nM T96413 CXD08L 155566182 IC50 = 28600 nM T04507 C91JWC 11619578 Ki = 16000 nM T04507 C9BN5X 25062886 Ki = 28000 nM T04507 C3JT6Y 25062887 Ki = 29000 nM T04507 C6FAE8 25128791 Ki = 950 nM T04507 C4LWD5 25133600 Ki = 8900 nM T04507 CI8QX9 25133601 Ki = 9300 nM T04507 CV74CM 25133602 Ki = 4200 nM T04507 C5SD4L 25133603 Ki = 4000 nM T04507 C34ICM 25133604 Ki = 1000 nM T04507 C5I9DS 25133605 Ki = 450 nM T04507 C8N4MR 25133945 Ki = 5200 nM T04507 C20HEP 25133946 Ki = 1600 nM T04507 CNZ57K 25133947 Ki = 2100 nM T04507 CB9S4K 25133948 Ki = 1100 nM T04507 CCH4Q7 25133949 Ki = 980 nM T04507 C1NE0M 44568787 Ki = 100000 nM T04507 C6O5MK 44568990 Ki = 78000 nM T04507 CBH3W2 44568992 Ki = 15000 nM T04507 CPE81S 44568993 Ki = 230000 nM T04507 CN8IJ2 44568997 Ki = 76000 nM T04507 CCZ07S 44568998 Ki = 29000 nM T04507 COQ86E 44569003 Ki = 67000 nM T04507 CBTY56 51349723 Ki = 110000 nM T04507 CLP7T1 51349724 Ki = 60000 nM T04507 C3W4VJ 51349725 Ki = 73000 nM T04507 C5V7FQ 51349853 Ki = 38000 nM T04507 CCK68B 51349854 Ki = 750 nM T04507 C9N3RK 51349855 Ki = 12000 nM T04507 C7M9VE 51349856 Ki = 4400 nM T04507 C4HCW7 51349857 Ki = 8100 nM T04507 CG6D0A 51349985 Ki = 3600 nM T04507 C2LED9 51349986 Ki = 1800 nM T04507 CM74JQ 51349987 Ki = 1200 nM T04507 CZC3I1 51349988 Ki = 56000 nM T04507 C8Q4JC 51349989 Ki = 13000 nM T04507 CS35NP 51350132 Ki = 1400 nM T04507 CB1FV4 51350133 Ki = 1200 nM T04507 CJ07LF 51350266 Ki = 1800 nM T04507 CK4LI9 51350267 Ki = 4200 nM T04507 C30CJU 51350268 Ki = 5000 nM T04507 C7FA1T 51350269 Ki = 9700 nM T04507 CA5KB6 51350401 Ki = 9000 nM T04507 C5BA4X 51350402 Ki = 16000 nM T04507 CSKF72 51350403 Ki = 33000 nM T04507 C0YT9S 51350544 Ki = 10800 nM T04507 CWC0V7 51350671 Ki = 220000 nM T04507 CL84AJ 51350797 Ki = 32000 nM T04507 C0KNX2 51350908 Ki = 630 nM T04507 CJD1A0 51350909 Ki = 1100 nM T04507 C1QND3 51350910 Ki = 1000 nM T04507 C0JTM6 53322961 Ki = 1500 nM T04507 C5Z4TK 53324180 Ki = 2100 nM T04507 C3NUX0 53324286 Ki = 22000 nM T04507 C3CG9X 53326546 Ki = 1300 nM T04507 CI4WU0 73350252 Ki = 2300 nM T04507 CYR89O 127045734 Ki = 229000 nM T04507 C3IGU0 127046244 Ki = 38000 nM T04507 C1NHQ9 127046286 Ki > 500000 nM T04507 CL47MV 127047627 Ki > 500000 nM T04507 C1YS3V 127047671 Ki = 530000 nM T04507 CZ0U9E 127047672 Ki = 289000 nM T04507 CE2N8U 127047673 Ki > 500000 nM T04507 D00SOE 44568937 Ki = 4100 nM T04507 D0UJ6V 44568938 Ki = 2100 nM T27445 D03JSJ 446596 Ki = 2.5 nM T27445 CP1ER7 10095725 Ki = 1.92 nM T27445 CO16MK 44287214 IC50 = 20 ug.mL-1 T27445 CATS31 44287256 IC50 = 9 ug.mL-1 T27445 C0HKM7 44287331 IC50 = 0.6 ug.mL-1 T27445 C5F8SW 44287472 IC50 = 289 ug.mL-1 T27445 CC2D4O 44287473 IC50 = 2.1 ug.mL-1 T27445 CUN84R 44287567 IC50 = 1.7 ug.mL-1 T27445 CKV87J 44287586 IC50 = 157 ug.mL-1 T27445 CNX61D 44287603 IC50 = 9.5 ug.mL-1 T27445 C71SKU 44287672 IC50 = 76 ug.mL-1 T27445 CTNX09 44287673 IC50 = 69 ug.mL-1 T27445 CHP85N 44287689 IC50 > 400 ug.mL-1 T27445 C1B6PL 44287840 IC50 = 0.1 ug.mL-1 T27445 CO9F8S 44288031 IC50 = 0.2 ug.mL-1 T27445 CS8U3V 44288047 IC50 > 400 ug.mL-1 T27445 CH81ZB 44288048 IC50 = 272 ug.mL-1 T27445 C0LB1H 44288049 IC50 = 0.85 ug.mL-1 T27445 C7XY4F 44385414 IC50 > 128000 nM T27445 CRB75J 44386149 IC50 > 128000 nM T27445 CQ9GZ3 44395765 IC50 = 6400 nM T27445 CF0Z5H 56671744 IC50 = 280000 nM T27445 C05DLC 56681810 IC50 = 35000 nM T27445 C9Z8RJ 71456287 IC50 = 19 ug.mL-1 T27445 CD1M7F 71461727 IC50 = 4.5 ug.mL-1 T27445 CE6G9D 90677447 Ki = 17.2 nM T27445 C80WRJ 90677448 Ki = 55 nM T27445 CJG28F 145971854 Ki = 213 nM T27445 C6W3XH 155537991 Ki = 1039 nM T27445 C53XCF 155556468 Ki = 1.2 nM T78127 D00KHM 16362 IC50 > 500000 nM T78127 D01AZG 5073 IC50 = 291000 nM T78127 D02DPA 2756 IC50 = 39000 nM T78127 D02PMO 60700 IC50 = 8600 nM T78127 D05DVP 5717 IC50 = 7600 nM T78127 D05EAM 4735 IC50 = 2700 nM T78127 D05HSC 6000 IC50 = 55500 nM T78127 D05PHH 3447 IC50 = 10800 nM T78127 D06NXY 5991 IC50 = 20200 nM T78127 D06ZUK 3696 IC50 > 100000 nM T78127 D07HOB 60838 IC50 = 7900 nM T78127 D0AV3G 3151 IC50 = 14800 nM T78127 D0AZ3C 5291 IC50 = 350 nM T78127 D0D9FV 4601 IC50 > 100000 nM T78127 D0DV3O 3241 IC50 = 29800 nM T78127 D0E6YQ 1935 IC50 > 100000 nM T78127 D0F9GE 3108 IC50 = 74000 nM T78127 D0H3HM 60795 IC50 > 500000 nM T78127 D0K0OZ 5702160 IC50 = 36200 nM T78127 D0K7WK 4595 IC50 = 160 nM T78127 D0M4YC 3114 IC50 > 100000 nM T78127 D0M7JT 216210 IC50 = 25300 nM T78127 D0NR6S 3002977 IC50 = 297000 nM T78127 D0R3JB 4212 IC50 = 530 nM T78127 D0T6XX 4679 IC50 = 43200 nM T78127 D0TQ1G 5071 IC50 = 288000 nM T78127 D0U2OO 2477 IC50 = 46000 nM T78127 D0V3ZA 10531 IC50 = 12600 nM T78127 D0V4GY 9552079 IC50 = 500 nM T78127 D0V7CF 5362440 IC50 = 7800 nM T78127 D0WV3U 4893 IC50 = 38400 nM T78127 D0ZU9R 392622 IC50 = 4400 nM T78127 D0Y6SQ 2536 IC50 = 12700 nM T78127 D0QQ1J 2406 IC50 = 6600 nM T78127 CP4RM6 4486 IC50 = 2700 nM T78127 CZA2C6 39764 IC50 = 25200 nM T78127 D0P2HR 3510 IC50 = 311000 nM T05904 D05MQK 110635 IC50 > 10000 nM T05904 D0Z7ZM 135398744 IC50 = 100000 nM T05904 D0T5PO 5092 IC50 > 16000 nM T05904 D0WS3T 72706254 IC50 = 8400 nM T05904 C8JLO0 2243267 IC50 > 10000 nM T05904 C45VZC 11438405 IC50 > 16000 nM T05904 CUK49V 11988837 Ki = 8200 nM T05904 CFIO49 11988967 Ki = 33000 nM T05904 C2D0NG 11989101 Ki = 54000 nM T05904 C65ABT 11989102 Ki > 100000 nM T05904 C1B4XD 11992634 IC50 > 2000 nM T05904 CPX16N 11993169 IC50 > 2000 nM T05904 C1PZ8C 18734933 IC50 > 16000 nM T05904 CW96SI 23624262 IC50 > 1000 nM T05904 C9WGI4 24802717 IC50 > 5000 nM T05904 C6EQG2 24963293 IC50 > 2000 nM T05904 CICF39 42629702 IC50 > 10000 nM T05904 CM3X9S 42629827 IC50 > 1000 nM T05904 CQN26J 42629945 IC50 > 10000 nM T05904 C6O5FX 42630062 IC50 > 10000 nM T05904 C71ZNR 42630180 IC50 > 10000 nM T05904 C4RHY0 42630191 IC50 > 10000 nM T05904 CT6RS9 42630192 IC50 > 10000 nM T05904 CYZL43 42630317 IC50 > 10000 nM T05904 CH42OZ 42630318 IC50 > 10000 nM T05904 C7X5AH 42630437 IC50 > 10000 nM T05904 CW8OB3 44243146 Ki > 10000 nM T05904 C5IMB2 46239424 Ki > 10000 nM T05904 CKR9P7 46239425 Ki > 10000 nM T05904 C3P2IN 46933992 IC50 >= 29000 nM T05904 CHA5Z0 49821469 IC50 > 1000 nM T05904 C1AYP0 49821627 IC50 > 500 nM T05904 C85AXR 49821714 IC50 > 1000 nM T05904 CEMS67 52938764 IC50 = 1.9 nM T05904 CT8FL5 54583590 IC50 = 1.8 nM T05904 CQC2V7 54584582 IC50 = 1.8 nM T05904 C8WH3R 54587529 IC50 = 1.8 nM T05904 CGF65A 54670110 IC50 > 30000 nM T05904 C90ZLC 54670399 IC50 > 30000 nM T05904 C4TGL7 56648496 IC50 > 1000 nM T05904 CH6C3L 56648679 IC50 > 10000 nM T05904 CCY79V 56648680 IC50 > 10000 nM T05904 CNE96P 56648857 IC50 > 10000 nM T05904 CX86AQ 56648859 IC50 > 5000 nM T05904 CPC3T4 56654131 IC50 > 10000 nM T05904 C0YD3P 56928304 IC50 > 5000 nM T05904 C8RO6A 56929788 IC50 > 1000 nM T05904 CD52CA 57391118 IC50 > 2000 nM T05904 CG3DF1 57392948 Ki > 10000 nM T05904 CE36TV 57394695 Ki > 10000 nM T05904 CPA3D1 57403394 Ki > 10000 nM T05904 C4XMB6 58547809 IC50 > 30000 nM T05904 CEB3G9 58547814 IC50 > 30000 nM T05904 C08QVG 58547833 IC50 > 30000 nM T05904 CFVG67 58547863 IC50 > 30000 nM T05904 CYZA38 58548077 IC50 > 30000 nM T05904 CC43LF 71074083 IC50 > 10000 nM T05904 C4P0XT 71092344 IC50 = 3560 nM T05904 C6DAG4 71092519 IC50 = 17000 nM T05904 C4GNJ3 71598545 IC50 > 1000 nM T05904 C7XRY6 72190879 IC50 > 30000 nM T05904 CQ3GD7 72704434 Ki = 3000 nM T05904 CF03DW 90168772 IC50 > 20000 nM T05904 CM6J9K 90168778 IC50 > 20000 nM T05904 CSCY01 117949009 IC50 > 10000 nM T05904 CYQ74R 118479645 IC50 > 10000 nM T05904 CVYK24 118556943 IC50 > 50000 nM T05904 CS6M9C 122193679 IC50 > 100000 nM T05904 C4UR7D 127038167 IC50 > 1000 nM T05904 C4H2TJ 127038168 IC50 > 1000 nM T05904 CL9JT8 127038169 IC50 > 1000 nM T05904 CJPX60 127038509 IC50 > 1000 nM T05904 C26EAG 127038511 IC50 > 1000 nM T05904 CTM9E4 127038512 IC50 > 1000 nM T05904 C6AQ2U 127038513 IC50 > 1000 nM T05904 CV1FM0 127038868 IC50 > 1000 nM T05904 CADU23 127038869 IC50 > 1000 nM T05904 CACJ46 132489333 IC50 = 6223 nM T05904 C2P1IU 134129996 IC50 > 100000 nM T05904 CLE03O 134130328 IC50 > 100000 nM T05904 CSN6J0 134130563 IC50 > 100000 nM T05904 C0A1CZ 134131162 IC50 > 100000 nM T05904 C3R8SE 135457869 IC50 > 10000 nM T05904 CHDC83 135566745 IC50 > 10000 nM T05904 C9IJK1 135566935 IC50 > 100000 nM T05904 CTX54Z 135896326 IC50 > 10000 nM T05904 C12UMG 136059728 IC50 > 1000 nM T05904 CRP24A 136087045 IC50 > 100000 nM T05904 C7SUX4 136087050 IC50 > 100000 nM T05904 C8UF7G 136087052 IC50 > 100000 nM T05904 C21FVA 136180322 IC50 > 10000 nM T05904 CQW7T0 136197286 IC50 > 10000 nM T05904 C8TQ7A 136217455 IC50 = 100000 nM T05904 C2N9VT 137348687 IC50 > 10000 nM T05904 C6KYD7 137700754 IC50 > 10000 nM T05904 CM3UF7 137700779 IC50 > 20000 nM T05904 CPTE92 138319693 IC50 > 32000 nM T05904 C2QLX3 138393292 IC50 > 50000 nM T05904 CMW20N 141737696 IC50 > 4000 nM T05904 C8HEG7 141737705 IC50 > 3000 nM T05904 CC7HN2 145974174 IC50 > 100000 nM T05904 CK1BR0 145978345 IC50 > 100000 nM T05904 CHJ79V 145997874 IC50 > 10000 nM T05904 CL8CU6 155521936 IC50 > 200000 nM T05904 CT85RG 155530589 IC50 > 200000 nM T05904 D09RKU 46239428 Ki > 10000 nM T05904 D0R6MT 3758 IC50 = 700000 nM T05904 D0V4WB 149790 IC50 > 16000 nM T26846 CL8RX5 1222 IC50 = 150000 nM T26846 CO9KU6 443586 EC50 = 65000 nM T26846 C6X8NA 44312783 EC50 > 300000 nM T26846 D04DKM 104766 EC50 = 50000 nM T12126 D03QLG 9917013 IC50 = 6 nM T12126 D0E3TC 44259 IC50 = 4 nM T12126 C8NW5J 3815 IC50 = 49 nM T12126 C9VW8M 449054 IC50 > 16000 nM T12126 C18WEB 490561 IC50 = 13 nM T12126 CK21EQ 9796713 IC50 = 40 nM T12126 CBT0X5 9797847 IC50 = 300 nM T12126 CJH69P 9840393 IC50 = 26 nM T12126 C7JE0V 9904731 IC50 = 277 nM T12126 CR3DA5 9939328 IC50 = 31 nM T12126 C6MO1K 10530175 IC50 = 11 nM T12126 CRJD61 10532168 IC50 = 94 nM T12126 CHB35P 10604501 IC50 = 143 nM T12126 C05KFQ 10604778 IC50 = 123 nM T12126 CJ4BN2 10626594 IC50 = 11 nM T12126 CGP93J 10745853 IC50 = 11 nM T12126 CO7Y9M 10770450 IC50 = 56 nM T12126 C7N2XF 10935867 IC50 = 270 nM T12126 CW3NL5 11012763 IC50 > 300 nM T12126 CD5I7L 11067837 IC50 = 58 nM T12126 CYXF06 11131268 IC50 = 171 nM T12126 CZ4F7B 11621437 IC50 = 20 nM T12126 C4NO7Y 11809063 IC50 = 87 nM T12126 C85WGB 12970028 IC50 = 1106 nM T12126 CAC69O 14677298 IC50 > 10000 nM T12126 CC3J9K 15736808 IC50 = 1200 nM T12126 C20DST 16105503 IC50 = 22 nM T12126 C47EWZ 16105505 IC50 > 300 nM T12126 CSQ86L 16105506 IC50 > 300 nM T12126 C28QKT 16105508 IC50 = 157 nM T12126 CXO3N2 16105509 IC50 = 110 nM T12126 CCN62F 16105510 IC50 = 12 nM T12126 C1JXQ8 16105511 IC50 = 724 nM T12126 C63QYN 16105513 IC50 > 300 nM T12126 CK0W9E 16105515 IC50 > 10000 nM T12126 C0USZ6 24971429 IC50 = 274 nM T12126 C8FK3N 24971430 IC50 = 159 nM T12126 C4LAW3 24971432 IC50 = 1000 nM T12126 C45WDR 24971433 IC50 = 87 nM T12126 C0B7RT 25057409 IC50 > 10000 nM T12126 CO42DC 44138048 IC50 > 10000 nM T12126 CL65QV 44138049 IC50 > 10000 nM T12126 C3E7RP 44284203 IC50 = 21 nM T12126 C8FY7N 44284204 IC50 = 44 nM T12126 CGC50I 44407533 IC50 > 1000 nM T12126 CU0H6W 44407571 IC50 > 1000 nM T12126 C3VRO9 44557921 IC50 > 10000 nM T12126 CC9X1M 46213938 IC50 = 78 nM T12126 CVJU38 46233842 IC50 = 19 nM T12126 CQ9A7L 46234188 IC50 = 7 nM T12126 C94GCA 46234349 IC50 = 9 nM T12126 C0AF2X 46234666 IC50 = 40 nM T12126 C9EMO2 54765177 IC50 = 21 nM T12126 CV63UL 67240318 IC50 > 10000 nM T12126 CZ4BX1 72547959 IC50 = 602 nM T12126 CQ2OB9 90292687 IC50 > 10000 nM T12126 CHI39S 90292823 IC50 > 10000 nM T12126 CJQ5N6 91936970 IC50 > 10000 nM T12126 C5N1VZ 102581295 IC50 > 10000 nM T12126 C2AN7T 134611886 IC50 > 100000 nM T12126 CGBZ13 134843302 IC50 = 500 nM T12126 C3MK9W 136807986 IC50 > 10000 nM T12126 CV9QD6 145968243 IC50 = 7 nM T12126 C68GMW 155538446 IC50 = 23000 nM T12126 CY6Q8S 155554337 IC50 = 19000 nM T12126 CO2I4P 155559898 IC50 = 600 nM T12126 D07ADX 54764565 IC50 = 14 nM T12126 D07IHM 9823787 IC50 = 65 nM T12126 D09QBA 23378546 IC50 = 55 nM T12126 D0N4LR 53469448 IC50 = 1140 nM T12126 D0YQ8V 46236221 IC50 = 3 nM T69200 CIPN50 71760902 IC50 > 1000 nM T69200 COZ8S1 78319129 IC50 > 1000 nM T69200 CW2VQ5 119058113 IC50 = 6200 nM T69200 CUWX94 119081692 IC50 = 9000 nM T69200 C3Q5GH 127048496 IC50 = 9600 nM T69200 CBIK03 127048805 IC50 = 11000 nM T69200 CVJ6I3 127049903 IC50 = 6900 nM T69200 C0OER5 127050110 IC50 = 7300 nM T69200 CIHP74 127050112 IC50 = 22000 nM T69200 CLQ5N2 134114171 IC50 = 1700 nM T69200 CV4X7R 135566898 Ki < 6560 nM T69200 CU2F1G 135566900 Ki < 6560 nM T69200 CW94QO 136226511 Ki < 6560 nM T69200 C6N4GP 137701967 IC50 < 5 nM T69200 CU0SA6 145978909 IC50 = 6 nM T69200 C5DGB8 145980671 IC50 = 570 nM T69200 CO9HF0 145981360 IC50 < 5 nM T69200 CGF0Y7 145982405 IC50 = 150 nM T69200 CQC67U 145986542 IC50 < 5 nM T69200 C42QNW 145988683 IC50 = 770 nM T69200 CSK4I3 145989316 IC50 = 30 nM T69200 CGA95I 145991552 IC50 = 30 nM T69200 C0W6CH 145992229 IC50 < 5 nM T69200 CM4W6U 145993894 IC50 = 10 nM T69200 D09HBR 135566899 Ki = 7970 nM T40694 D01ZRI 6450551 IC50 > 10000 nM T40694 D07POC 176870 IC50 > 100000 nM T40694 D08CDI 208908 IC50 > 100000 nM T40694 D0K8KX 5280343 IC50 = 5750 nM T40694 D0R0MW 5329102 IC50 > 10000 nM T40694 D00BYM 10461508 IC50 = 0.87 nM T40694 D02KKA 24856436 IC50 = 350 nM T40694 D02RJY 11442891 IC50 = 3500 nM T40694 D02UFQ 11620908 IC50 > 10000 nM T40694 D02ZQS 16095342 IC50 > 10000 nM T40694 D03HUX 49792852 IC50 = 2 nM T40694 D03LWG 53235510 IC50 > 10000 nM T40694 D07EHV 44814409 IC50 > 10000 nM T40694 D07HPJ 11476171 IC50 > 10000 nM T40694 D08RMJ 15983966 Ki = 2.2 nM T40694 D09JGK 53357478 IC50 = 2 nM T40694 D0A5MC 11712649 IC50 = 53000 nM T40694 D0CY1B 6420138 Ki > 10000 nM T40694 D0E3TC 44259 IC50 = 0.92 ug.mL-1 T40694 D0KF9Q 6918736 IC50 = 9 nM T40694 D0O0LQ 11364421 Ki = 0.22 nM T40694 D0O0LS 25141092 IC50 > 10000 nM T40694 D0O6WV 24794418 IC50 > 2000 nM T40694 D0P1CV 46191454 IC50 > 10000 nM T40694 D0Q7RE 16007391 Ki > 10000 nM T40694 D0Q9UX 16718576 IC50 > 10000 nM T40694 D03BNU 59604787 IC50 > 10000 nM T40694 D05ZCQ 9548005 IC50 = 900 nM T40694 D00PWQ 3820 IC50 > 100000 nM T40694 D09SFV 3973 IC50 = 2000 nM T40694 D0P1JI 312145 IC50 = 5.8 nM T40694 D0T3ME 156422 IC50 > 30000 nM T40694 C3ZVJ9 10281 IC50 = 2180 nM T40694 C63WLY 89644 IC50 = 4.8 ug.mL-1 T40694 C5JE2Z 104860 IC50 > 10 ug.mL-1 T40694 CI1NA5 159926 IC50 > 10 ug.mL-1 T40694 CYBA43 177458 IC50 > 10 ug.mL-1 T40694 CN05AH 406563 IC50 > 10000 nM T40694 CXS8U2 447960 IC50 = 10000 nM T40694 CB9F1O 447961 Ki > 1000 nM T40694 C1ZG2U 449087 IC50 > 10000 nM T40694 CUO5Y3 1020400 IC50 > 10000 nM T40694 C3L7YE 2077962 IC50 = 25000 nM T40694 CIHY32 2190510 IC50 = 3200 nM T40694 C4D0HJ 2779943 IC50 = 56000 nM T40694 C86LNP 2779952 IC50 = 500 nM T40694 CVZ9D0 3162171 IC50 = 3 nM T40694 C8IAR2 5281657 IC50 = 75700 nM T40694 CI68PW 5283685 IC50 > 100000 nM T40694 CXK0S6 5283727 IC50 > 100000 nM T40694 CDQ3M7 5359485 IC50 = 6.9 ug.mL-1 T40694 C54BYP 5360741 IC50 = 8.2 ug.mL-1 T40694 C36GHS 5735633 IC50 > 10000 nM T40694 CT8U7I 5874584 IC50 = 25000 nM T40694 C34FPE 6510285 IC50 = 29000 nM T40694 CM35CV 6539291 IC50 = 5000 nM T40694 CT7MP9 6539292 IC50 = 25000 nM T40694 CKIP13 7769752 IC50 = 3600 nM T40694 C4G9WR 9547398 IC50 > 100000 nM T40694 C76CUP 9547698 IC50 > 100000 nM T40694 CCIP93 9548007 IC50 = 8000 nM T40694 CQ57EC 9548013 IC50 = 20 nM T40694 C3YDS0 9613592 IC50 = 29400 nM T40694 C9TAL6 9826308 IC50 = 2 nM T40694 CW8V0K 9864418 IC50 > 25000 nM T40694 CSL50Q 9886746 IC50 = 40 nM T40694 CJ03FO 9891182 Ki = 12 nM T40694 C4WSV3 9906179 IC50 = 580 nM T40694 CS5KX9 9938299 IC50 > 10000 nM T40694 CS23WF 9983158 IC50 = 5 nM T40694 C37GXK 9983303 IC50 > 25000 nM T40694 CR8DA1 10024683 IC50 > 100000 nM T40694 CLA93G 10047202 IC50 = 100000 nM T40694 C3LCH5 10047545 IC50 > 100000 nM T40694 C40TGW 10074495 IC50 = 12 nM T40694 CD6V3C 10085550 IC50 = 21000 nM T40694 C2C1BP 10089048 IC50 > 25000 nM T40694 CGT7V4 10216158 IC50 = 10000 nM T40694 CPK70Y 10253033 IC50 = 2 nM T40694 CVW4N2 10254917 IC50 = 2 nM T40694 C3FR5E 10401406 IC50 = 39000 nM T40694 CBJ3F6 10409707 EC50 = 2000 nM T40694 C4CP7K 10423452 IC50 = 8800 nM T40694 C7HBP6 10429593 IC50 > 10000 nM T40694 CRX6F0 10479082 IC50 > 25000 nM T40694 CEML49 10538870 IC50 > 100000 nM T40694 C9O2PG 10588346 IC50 > 100000 nM T40694 C7BK0W 10635986 Ki > 44000 nM T40694 C7KF2E 10705154 IC50 > 100000 nM T40694 C83QWV 10714343 IC50 = 21700 nM T40694 C2C8GH 10732141 IC50 > 100000 nM T40694 C16DOZ 10849808 Ki = 32000 nM T40694 CC0OD9 11155941 IC50 = 500 nM T40694 CJ7U4I 11161778 IC50 < 50000 nM T40694 CNI7Q5 11174936 IC50 = 300 nM T40694 CW8K1B 11185889 IC50 > 10000 nM T40694 C9Y1GN 11187801 IC50 > 10000 nM T40694 CU50CB 11189040 IC50 = 80 nM T40694 C8G5WP 11210533 IC50 = 6310 nM T40694 CTK8R1 11211191 IC50 = 2740 nM T40694 C7VRB8 11213555 IC50 = 70 nM T40694 C1IM0Q 11244902 IC50 = 2810 nM T40694 C0BW3Q 11260691 IC50 = 1.1 nM T40694 C6C3JX 11281930 IC50 > 10000 nM T40694 CMJ01U 11283298 IC50 = 9 nM T40694 CEJ96I 11293491 IC50 = 1980 nM T40694 CBOP58 11293798 Ki = 1280 nM T40694 CPTO12 11294348 IC50 = 2670 nM T40694 C3F6UB 11300082 IC50 = 1131 nM T40694 CX45OL 11304724 IC50 = 5660 nM T40694 C0FS8C 11328632 IC50 = 30 nM T40694 C26BZX 11362471 Ki = 940 nM T40694 C4T5KR 11372661 IC50 = 380 nM T40694 CWXB93 11397177 Ki = 2330 nM T40694 CEN76S 11405758 IC50 = 90 nM T40694 CB96XY 11438062 IC50 = 1200 nM T40694 C8KSH5 11465304 IC50 = 1060 nM T40694 C4YVO2 11466081 IC50 = 410 nM T40694 C9LA1E 11486283 IC50 > 10000 nM T40694 C8I1JT 11495629 IC50 = 7.3 nM T40694 C21NXF 11500264 IC50 = 13700 nM T40694 C68TQO 11502143 IC50 = 31 nM T40694 C5R3WT 11522898 IC50 = 6500 nM T40694 CL7X4Q 11530963 IC50 > 100000 nM T40694 CTG83F 11539329 Ki > 8900 nM T40694 CG17OP 11572678 IC50 = 7800 nM T40694 CRZJ71 11580497 IC50 = 8700 nM T40694 C75MUQ 11587793 IC50 = 6900 nM T40694 CMIL86 11590363 Ki > 8900 nM T40694 CO2JL0 11625181 IC50 < 10000 nM T40694 CSM62L 11626920 IC50 > 30000 nM T40694 CGX96V 11626927 IC50 = 794.33 nM T40694 C9T6SC 11640926 Ki > 8900 nM T40694 C4GTZ8 11645322 IC50 > 20000 nM T40694 CE80VT 11656480 EC50 = 19000 nM T40694 CZE9U8 11661872 EC50 = 80 nM T40694 CU0E8O 11690457 Ki > 10000 nM T40694 C0CE3I 11698712 EC50 = 48000 nM T40694 CB0AP2 11705863 Ki > 4000 nM T40694 CJ9FB6 11743086 IC50 = 21 nM T40694 CVFS29 11751305 IC50 = 530 nM T40694 C9JT4S 11847343 IC50 > 10000 nM T40694 CW3K2L 11957417 IC50 = 0.8 nM T40694 CDGF78 15282555 IC50 = 3900 nM T40694 CFPW41 16007116 Ki > 8900 nM T40694 CT37CO 16050921 IC50 = 3 nM T40694 CW2XK6 16050925 IC50 = 2 nM T40694 CZHJ34 16058637 IC50 = 730 nM T40694 C7Z4LV 16095343 IC50 > 10000 nM T40694 CU56EW 16664858 IC50 > 10000 nM T40694 CD6Z8F 16722190 IC50 = 12 nM T40694 C9IW5S 16730105 IC50 = 5700 nM T40694 CA61QF 21083895 IC50 < 50000 nM T40694 CL81VC 21100709 IC50 = 100000 nM T40694 C6Y1BF 23624256 Ki = 234 nM T40694 CYM03F 24281531 IC50 = 31 nM T40694 C7YG1N 24759534 IC50 = 55000 nM T40694 CCPS81 24764502 IC50 > 35000 nM T40694 CJUK39 24770517 IC50 > 10000 nM T40694 C35JHQ 24812745 IC50 = 3 nM T40694 CCP2M3 24822704 IC50 > 50000 nM T40694 C5YW7P 24825755 IC50 = 3 nM T40694 C61KPI 24856363 IC50 > 25000 nM T40694 CRQJ49 24864675 Ki = 354 nM T40694 C2VQC5 24864676 Ki = 9930 nM T40694 CAR4Y8 24864677 Ki = 272 nM T40694 CX4I2B 24864678 Ki = 465 nM T40694 C81OJV 24864855 Ki = 771 nM T40694 C6UOY5 24865032 Ki = 141 nM T40694 C0QC1S 24865034 Ki = 610 nM T40694 CTM2N6 24875313 IC50 = 720 nM T40694 C13QYB 24884503 IC50 > 2000 nM T40694 CN13JF 24899915 IC50 = 4.4 ug.mL-1 T40694 CBWR97 24899916 IC50 = 5.7 ug.mL-1 T40694 C9F2JD 24899917 IC50 > 10 ug.mL-1 T40694 C64MTI 24900160 IC50 > 10 ug.mL-1 T40694 CO2I6Q 24900161 IC50 > 10 ug.mL-1 T40694 C7B8NG 24941248 IC50 = 99 nM T40694 CJ43DG 24954671 IC50 = 1 nM T40694 C4V9GI 24960018 IC50 > 50000 nM T40694 CVOU94 24971414 IC50 = 1301 nM T40694 CYOA93 24971415 IC50 = 121 nM T40694 C03UHR 24971416 IC50 = 1616 nM T40694 C7PYN2 24971417 IC50 = 549 nM T40694 CQZ6M1 24971418 IC50 = 1170 nM T40694 C9JKR8 24971419 IC50 = 330 nM T40694 C5V0DH 24971420 IC50 = 625 nM T40694 CE4HL7 24971421 IC50 = 4927 nM T40694 CN1D2A 24971422 IC50 = 214 nM T40694 C3LOR9 24971423 IC50 = 51 nM T40694 CSHX05 24971424 IC50 > 20000 nM T40694 CVO16F 24971425 IC50 = 3007 nM T40694 CTM6Y7 24971426 IC50 = 779 nM T40694 CYU62O 24971427 IC50 = 5689 nM T40694 C32SIZ 24971428 IC50 = 7479 nM T40694 CQEV29 24992861 IC50 = 15 nM T40694 CCZF80 24992862 IC50 = 110 nM T40694 CU5B6R 24992864 IC50 = 109 nM T40694 C4EG8R 24993189 IC50 = 7 nM T40694 CS3Q8B 24995659 Ki > 4000 nM T40694 CBK82P 25011729 IC50 > 30000 nM T40694 CX1HL8 25032704 Ki > 8890 nM T40694 C0B7RT 25057409 IC50 > 10000 nM T40694 CC3SM2 25093244 IC50 = 7685 nM T40694 C6BAW9 25093245 IC50 = 474 nM T40694 C1M9AD 25093246 IC50 = 4528 nM T40694 C05ZXF 25093247 IC50 = 14451 nM T40694 CKV73D 25093248 IC50 = 5928 nM T40694 C8VPB5 25093249 IC50 = 703 nM T40694 CHIW69 25093250 IC50 = 4516 nM T40694 CR7E8V 25093251 IC50 = 464 nM T40694 CUA0G2 25093252 IC50 = 3241 nM T40694 CTDK51 25093253 IC50 = 1476 nM T40694 CXP4J0 25093254 IC50 = 412 nM T40694 CI47VM 25093255 IC50 = 977 nM T40694 C15EUS 25093256 IC50 = 225 nM T40694 C4ZO3U 25093257 IC50 = 149 nM T40694 CA9M5H 25093258 IC50 = 641 nM T40694 C2N3RP 25093259 IC50 = 274 nM T40694 C3L0EN 25093260 IC50 = 21 nM T40694 C3TF9O 25093261 IC50 = 32 nM T40694 CI1MK8 25093262 IC50 = 48 nM T40694 C49SOI 25093263 IC50 = 59 nM T40694 CES32T 25093264 IC50 = 207 nM T40694 CIG4H0 25178539 IC50 = 9900 nM T40694 CPL20E 25190911 IC50 = 70 nM T40694 CF4H8C 25190912 IC50 = 75 nM T40694 CYG76T 25190913 IC50 = 630.96 nM T40694 CMQ32Y 25190914 IC50 = 251.19 nM T40694 C2RYF9 25190915 IC50 = 700 nM T40694 CNG96H 25210579 IC50 = 9 nM T40694 CCDT62 25252909 IC50 = 2 nM T40694 C8UT3C 25252911 IC50 = 100 nM T40694 CD7HY1 25253225 IC50 = 5 nM T40694 CAJR97 25253226 IC50 = 170 nM T40694 CQB7W4 25253376 IC50 = 3 nM T40694 C8AC2D 25253525 IC50 = 1 nM T40694 C1YNQ8 25263074 IC50 = 61 nM T40694 CN7TD8 25263075 IC50 = 12 nM T40694 C69QGA 25263076 IC50 = 12 nM T40694 CPB62E 25263077 IC50 = 12 nM T40694 C2M9SZ 25263078 IC50 = 28 nM T40694 CRK3L4 25263079 IC50 = 35 nM T40694 C2E6BO 25263080 IC50 = 12 nM T40694 CM6TK2 25263081 IC50 = 22 nM T40694 C01RET 25263082 IC50 = 100 nM T40694 CM4U0X 25263083 IC50 = 11 nM T40694 C0WH3J 25263084 IC50 = 14 nM T40694 CP7WG9 25263085 IC50 = 21 nM T40694 C1D8VW 25263086 IC50 = 4 nM T40694 CSKW68 25263087 IC50 = 300 nM T40694 CXKJ04 25263089 IC50 = 250 nM T40694 CDX5G1 25263090 IC50 = 8 nM T40694 CUZ9A7 25263091 IC50 = 12 nM T40694 CBJ06W 25263092 IC50 = 2 nM T40694 C0KAU6 25263093 IC50 = 6 nM T40694 CA6TJ8 25263094 IC50 = 17 nM T40694 C7MDF9 25263095 IC50 = 8 nM T40694 CU7Q6Y 25263096 IC50 = 31 nM T40694 CI5W1P 25263097 IC50 = 99 nM T40694 C9H5ED 25263098 IC50 = 13 nM T40694 CF46NW 25263099 IC50 = 130 nM T40694 CGRW37 25263100 IC50 = 61 nM T40694 C91MSJ 25263101 IC50 = 34 nM T40694 C98RJP 25263102 IC50 = 17 nM T40694 CLM4E7 25263103 IC50 = 11 nM T40694 CH4E9T 25263104 IC50 = 17 nM T40694 C5CK0G 25263105 IC50 = 2 nM T40694 C50XJV 25263106 IC50 = 27 nM T40694 CC75GK 25263107 IC50 = 190 nM T40694 CA2O1W 25263108 IC50 = 130 nM T40694 C6LD1H 25263109 IC50 = 14 nM T40694 CJGD56 25263110 IC50 > 1000 nM T40694 CQ60NP 25263111 IC50 = 2 nM T40694 C51DJI 25263112 IC50 = 73 nM T40694 CUJM96 25263113 IC50 = 6 nM T40694 CT1L6J 25263114 IC50 = 85 nM T40694 CM45AK 25263115 IC50 > 1000 nM T40694 CIM8G1 25263116 IC50 > 1000 nM T40694 CDS1I3 25263117 IC50 = 30 nM T40694 CUK69B 25263118 IC50 = 1 nM T40694 CX06UC 25263119 IC50 = 3 nM T40694 CY87ZW 25263120 IC50 = 1 nM T40694 C4YVP3 25263121 IC50 = 4 nM T40694 C85UOW 25263123 IC50 = 7 nM T40694 CH7WZ5 25263124 IC50 = 6 nM T40694 CLDB65 25263125 IC50 = 3 nM T40694 C3CK5M 25263126 IC50 = 4 nM T40694 CN5E0F 25263283 IC50 = 12000 nM T40694 CU53WB 42596953 IC50 = 6800 nM T40694 CX03BO 42608451 IC50 = 5270 nM T40694 CJ5U1X 42639664 IC50 > 10 ug.mL-1 T40694 C2CTI1 44129603 IC50 = 110 nM T40694 CO42DC 44138048 IC50 > 10000 nM T40694 CL65QV 44138049 IC50 > 10000 nM T40694 C8KNA3 44219632 Ki > 4000 nM T40694 C0VIX4 44219633 Ki > 4000 nM T40694 CEL61X 44229839 IC50 > 10000 nM T40694 C6G2EC 44232693 IC50 > 10000 nM T40694 CGTI98 44232942 IC50 > 10000 nM T40694 CCG09Z 44235884 IC50 > 10000 nM T40694 C13QXB 44236351 IC50 = 68 nM T40694 CJ37DI 44236353 IC50 = 4215 nM T40694 CGI5L7 44405938 IC50 > 20000 nM T40694 C0G3WF 44405939 IC50 > 20000 nM T40694 CR3Q7Z 44405940 IC50 > 20000 nM T40694 C79WRL 44405941 IC50 = 16000 nM T40694 C9ZNA0 44405945 IC50 > 100000 nM T40694 C9LD2T 44405946 IC50 > 100000 nM T40694 C0RO6U 44405949 IC50 > 20000 nM T40694 C2CTN7 44405982 IC50 > 100000 nM T40694 C0CR1O 44405983 IC50 = 21000 nM T40694 CW86VI 44405987 IC50 > 100000 nM T40694 C5V4TQ 44405999 IC50 = 23000 nM T40694 C0XZ8K 44406013 IC50 = 17000 nM T40694 CS3K1P 44406014 IC50 > 20000 nM T40694 CC93JP 44406018 IC50 > 20000 nM T40694 C7P0IH 44406019 IC50 > 20000 nM T40694 C4X2ME 44406047 IC50 = 8000 nM T40694 C36YDV 44406048 IC50 > 100000 nM T40694 CXZ5C3 44406055 IC50 > 100000 nM T40694 CCRZ12 44406074 IC50 = 12000 nM T40694 CHR6A1 44420293 IC50 = 630.96 nM T40694 COPG94 44427519 IC50 > 10000 nM T40694 CZ1R8M 44450033 IC50 > 100000 nM T40694 CIY3T5 44450035 IC50 > 100000 nM T40694 C5Y4PN 44450059 IC50 = 50000 nM T40694 C28LMV 44450060 IC50 > 100000 nM T40694 C97CDF 44555517 IC50 > 10000 nM T40694 CY2GA6 44555518 IC50 > 10000 nM T40694 CPV8A6 44555519 IC50 > 10000 nM T40694 C9Q8VR 44555761 IC50 > 10000 nM T40694 C68LVU 44555820 IC50 > 10000 nM T40694 CP6FY8 44556163 IC50 = 237 nM T40694 CHA25B 44556214 IC50 = 3034 nM T40694 CR2CH3 44556329 IC50 = 1652 nM T40694 CN94PG 44578858 IC50 = 23 nM T40694 CE06BJ 44578859 IC50 = 34 nM T40694 CE2JI4 44578906 IC50 = 41 nM T40694 CI6O0P 44579005 IC50 = 71 nM T40694 CS9QC2 44579006 IC50 = 74 nM T40694 CQ13WT 44579007 IC50 = 100 nM T40694 C3O1EK 44579008 IC50 = 160 nM T40694 C6HY9O 44579009 IC50 = 270 nM T40694 CR1BW5 44579061 IC50 = 330 nM T40694 C4BA2J 44579062 IC50 = 550 nM T40694 C6HAE2 44579063 IC50 = 750 nM T40694 CPVK67 44579103 IC50 = 960 nM T40694 CAT3Y9 44579104 IC50 = 1040 nM T40694 C6JXV0 44579148 IC50 = 36 nM T40694 CHDW32 44579149 IC50 = 37 nM T40694 C8BCZ2 44579150 IC50 = 46 nM T40694 CDUM18 44579203 IC50 = 81 nM T40694 C9V4BU 44579204 IC50 = 190 nM T40694 C9B7FO 44579205 IC50 = 345 nM T40694 CAP6B1 44579206 IC50 = 490 nM T40694 CRFJ49 44579245 IC50 = 500 nM T40694 CZH86I 44579246 IC50 = 1600 nM T40694 CZIS45 44579247 IC50 = 1600 nM T40694 C7Q1VU 44580077 IC50 > 25000 nM T40694 CL90SE 44580358 IC50 > 25000 nM T40694 CK1VE7 44580420 IC50 > 25000 nM T40694 CH2R7X 44580449 IC50 > 25000 nM T40694 C1VH0C 44580532 IC50 > 25000 nM T40694 CXC52J 44580649 IC50 > 25000 nM T40694 CV49RU 44580656 IC50 = 42 nM T40694 C3FX7B 44580657 IC50 = 50 nM T40694 CE32BQ 44580689 IC50 > 25000 nM T40694 C8Z5AX 44580778 IC50 > 25000 nM T40694 CIB1C2 44589693 IC50 = 1500 nM T40694 C8YKG9 44589694 IC50 > 10000 nM T40694 C9PLW6 44589695 IC50 > 10000 nM T40694 CB5FN6 44589696 IC50 > 10000 nM T40694 C4Z7FI 44589729 IC50 = 680 nM T40694 CM79CZ 44634484 IC50 = 3.9 nM T40694 CU3RF1 45139989 IC50 > 10000 nM T40694 CQGZ06 45139991 IC50 > 10000 nM T40694 CST89M 45267711 EC50 = 290000 nM T40694 CUZ05J 45267745 IC50 = 130 nM T40694 CSQM53 45267772 IC50 = 12 nM T40694 C9T5YI 45268586 IC50 = 210 nM T40694 CS38DX 45269431 IC50 = 13 nM T40694 C8R7PS 45269486 EC50 = 310 nM T40694 C0PJ2H 45269487 IC50 = 88 nM T40694 CO1M5E 45269500 EC50 = 68000 nM T40694 C9GP3B 45269501 IC50 = 25 nM T40694 C4LQ5Z 45269507 EC50 = 184000 nM T40694 C4W1UX 45269647 IC50 > 10000 nM T40694 COB5N6 45270331 IC50 = 92 nM T40694 CJZT14 45270344 EC50 = 120000 nM T40694 C4YN1D 45271090 IC50 = 12 nM T40694 C5BMQ9 45271099 IC50 = 20 nM T40694 CIN3Q5 45271158 EC50 = 36000 nM T40694 C0GLX2 45271161 EC50 = 37000 nM T40694 CO4K6N 45271168 EC50 = 219000 nM T40694 C2YLW6 45271969 EC50 = 390000 nM T40694 C26ZVG 45271970 EC50 = 227000 nM T40694 CXR3W7 45271975 IC50 = 16 nM T40694 CG51PM 45272047 IC50 > 3000 nM T40694 CMF09J 45272048 IC50 > 3000 nM T40694 C2TD6R 45272052 IC50 = 300 nM T40694 CKG32D 45272066 IC50 = 22 nM T40694 CCQH35 45272865 IC50 = 430 nM T40694 C96YKJ 45272866 IC50 = 2100 nM T40694 CA05ZQ 45273759 IC50 = 17 nM T40694 C2B6VZ 45273767 IC50 = 150 nM T40694 CMI49Y 45273806 EC50 = 5000 nM T40694 CT4G1X 45273808 IC50 = 35 nM T40694 CL9X0C 45273817 EC50 = 1160 nM T40694 C2C8RH 45379202 IC50 > 100000 nM T40694 C5NB2X 45379203 IC50 > 100000 nM T40694 CT5BJ1 45379204 IC50 > 100000 nM T40694 CB41VP 45379205 IC50 > 100000 nM T40694 C2VUR3 45379340 IC50 > 100000 nM T40694 C8WXT4 45379341 IC50 > 100000 nM T40694 CQL29T 45379342 IC50 > 100000 nM T40694 CM7CB1 45379343 IC50 > 100000 nM T40694 C68WYX 45379344 IC50 > 100000 nM T40694 C27MFU 45379345 IC50 = 15000 nM T40694 C2O6VB 45379346 IC50 = 47000 nM T40694 CLMB07 45379347 IC50 > 100000 nM T40694 C8H5BL 45379490 IC50 > 100000 nM T40694 C4YV6H 45379491 IC50 > 100000 nM T40694 CRK4H3 45379492 IC50 > 100000 nM T40694 CSM20A 45379493 IC50 > 100000 nM T40694 CWP35H 45379494 IC50 > 100000 nM T40694 CV2AZ7 45379495 IC50 = 19000 nM T40694 CMP03L 45379496 IC50 = 73000 nM T40694 C6HM4U 45379605 IC50 > 100000 nM T40694 C6T1SW 45379606 IC50 = 14000 nM T40694 CHNS21 45379607 IC50 = 9300 nM T40694 C8HV1P 45379608 IC50 = 20000 nM T40694 CT6U7X 45379609 IC50 = 350 nM T40694 C5ATD8 45379610 IC50 = 750 nM T40694 C2APY4 45379611 IC50 = 7300 nM T40694 CODU08 45379711 IC50 = 840 nM T40694 C79MTY 45379712 IC50 = 140 nM T40694 C8LMI5 45379713 IC50 = 360 nM T40694 CTJQ49 45379714 IC50 = 2500 nM T40694 C15CVY 45379715 IC50 = 2600 nM T40694 CM0P8B 45379716 IC50 = 1700 nM T40694 C9XC4B 45379717 IC50 = 2300 nM T40694 C1U6ST 45379811 IC50 = 1400 nM T40694 CWB1C2 45379812 IC50 > 100000 nM T40694 CATM81 45379814 IC50 > 100000 nM T40694 C4W3OR 45379815 IC50 > 100000 nM T40694 C7NY4T 46223562 IC50 = 6 nM T40694 CG1H6A 46223563 IC50 > 10000 nM T40694 CK4W3S 46223564 IC50 = 248 nM T40694 CGNY46 46223565 IC50 = 143 nM T40694 C0OG3H 46223566 IC50 = 430 nM T40694 CG18LT 46223796 IC50 > 10000 nM T40694 CEJ1G8 46223797 IC50 > 10000 nM T40694 CY3HW5 46224684 IC50 > 10000 nM T40694 C7ON5A 46233287 IC50 > 10000 nM T40694 C9H4YO 46233889 EC50 = 33000 nM T40694 CRT34L 46235770 IC50 = 1 nM T40694 CLS29B 46872626 IC50 > 10000 nM T40694 C2O8RZ 46886323 IC50 > 1000 nM T40694 C5M8UY 46886877 IC50 = 432 nM T40694 C6XIZ3 46886878 IC50 = 51 nM T40694 CQI12F 46886956 IC50 = 872 nM T40694 C3RIH2 46886957 IC50 = 346 nM T40694 CZ4J8I 46886958 IC50 = 100 nM T40694 CBJ26E 46886959 IC50 = 197 nM T40694 CMU45C 46886960 IC50 = 42 nM T40694 C38MVY 46887029 IC50 = 135 nM T40694 C3Y5NA 46887030 IC50 = 256 nM T40694 C1SJ7I 46887031 IC50 = 488 nM T40694 C32MST 46887032 IC50 > 10000 nM T40694 CN4O5T 46887033 IC50 > 10000 nM T40694 C7JG4Q 46887069 IC50 = 97 nM T40694 CYG3B2 46887070 IC50 = 125 nM T40694 C82SLV 46887071 IC50 = 365 nM T40694 CD4Y9O 46887101 IC50 = 1117 nM T40694 CYL4K8 46887102 IC50 = 2076 nM T40694 C29OLT 46887103 IC50 = 3733 nM T40694 CW5P4R 46887104 IC50 = 1565 nM T40694 C1W3QP 46887105 IC50 = 278 nM T40694 CJ0QH7 46887137 IC50 = 943 nM T40694 C8GO5N 46887138 IC50 = 949 nM T40694 CL5IQ9 46887139 IC50 = 1969 nM T40694 CFV71W 46887140 IC50 = 2033 nM T40694 C45OAG 46887187 IC50 = 150 nM T40694 CW13FN 46887188 IC50 = 2523 nM T40694 C5X8BP 46887189 IC50 = 2051 nM T40694 CB8Q1F 46887190 IC50 = 464 nM T40694 CK1YB8 46887222 IC50 = 40 nM T40694 C5G2VE 46909588 IC50 > 5000 nM T40694 CH30UW 46911118 IC50 = 1 nM T40694 C4WXU5 46911119 IC50 = 1 nM T40694 C2YM9P 46911173 IC50 = 1 nM T40694 CZ3XP5 46926535 IC50 = 22600 nM T40694 C60GAV 46929544 IC50 > 8000 nM T40694 CP34VL 46929748 IC50 > 1000 nM T40694 CJ2E9Q 46929857 IC50 > 25000 nM T40694 CHSF07 49806372 IC50 > 1000 nM T40694 C75GBE 49837568 IC50 = 8500 nM T40694 C9L3XR 49838879 IC50 > 15000 nM T40694 CF91RS 49843531 IC50 > 10000 nM T40694 CE7D2J 49855568 IC50 = 12000 nM T40694 CFD9P3 49855569 IC50 = 2700 nM T40694 C1AU5N 49855758 IC50 = 9100 nM T40694 CIFK93 49855759 IC50 = 3900 nM T40694 CK48OJ 49855760 IC50 = 5600 nM T40694 CZI3M1 49855761 IC50 = 8500 nM T40694 CRPZ58 49855949 IC50 = 5500 nM T40694 CTU0K3 49855950 IC50 = 6200 nM T40694 CF85NL 49855951 IC50 = 27000 nM T40694 CF7YS9 49855952 IC50 = 2000 nM T40694 CJU38G 49855953 IC50 = 2900 nM T40694 CD95IE 49862008 IC50 = 4 nM T40694 C8GUQ2 49862009 IC50 = 53 nM T40694 CXT41G 49862010 IC50 = 1 nM T40694 COS71Z 49862053 IC50 = 1 nM T40694 C8D5XS 49862054 IC50 = 1 nM T40694 CPL5O8 49862055 IC50 = 8 nM T40694 C2H9XC 49862090 IC50 = 2 nM T40694 C4RNH2 49862091 IC50 = 3 nM T40694 CY9QB4 49862092 IC50 = 5 nM T40694 CC6NY3 49862093 IC50 = 1 nM T40694 C6MP7Y 49862094 IC50 = 2 nM T40694 CK8M2Y 49862095 IC50 = 1 nM T40694 CDK7E2 49862126 IC50 = 1 nM T40694 CKO54S 49862127 IC50 = 1 nM T40694 C3O5IR 49862128 IC50 = 2 nM T40694 CK72LH 49862588 IC50 = 6 nM T40694 CVN91K 49862589 IC50 = 18 nM T40694 C87LOT 49862590 IC50 = 1 nM T40694 CZ93HB 49862591 IC50 = 2 nM T40694 CI41BU 49862643 IC50 = 1 nM T40694 C1WXU4 49862644 IC50 = 2 nM T40694 C1W0AU 49862645 IC50 = 1 nM T40694 C7RCS0 49862646 IC50 = 2 nM T40694 C8L4QS 49862708 IC50 = 6 nM T40694 C2MT4B 49862709 IC50 = 3 nM T40694 CC5G9Y 49862710 IC50 = 5 nM T40694 CH5R7F 49862711 IC50 = 1 nM T40694 C10CAN 49862783 IC50 = 1 nM T40694 C4IH1S 49862784 IC50 = 1 nM T40694 CJTY17 49862785 IC50 = 1 nM T40694 CT81YB 49873221 IC50 = 16000 nM T40694 CBC62W 50899254 IC50 = 2 nM T40694 CD2K4R 50908681 IC50 = 271000 nM T40694 C2Y6QS 50938552 IC50 > 10000 nM T40694 CN4F3J 50990893 IC50 < 9 nM T40694 CLO87M 50990894 IC50 = 51300 nM T40694 C9NYP4 51036677 IC50 > 10000 nM T40694 C4WRY3 51037112 IC50 > 10000 nM T40694 CRI28Z 51037948 IC50 > 10000 nM T40694 C9MF0X 51355153 IC50 = 69 nM T40694 COR06H 51355154 IC50 = 66 nM T40694 C5E7UN 51355155 IC50 = 1330 nM T40694 CPLQ60 51355435 IC50 = 5310 nM T40694 CWJ46U 51355436 IC50 < 9 nM T40694 CF1D9W 51355713 IC50 = 87900 nM T40694 CDT46W 51355977 IC50 = 15200 nM T40694 CZ82JE 51357926 IC50 = 190 nM T40694 CM24LF 52938983 IC50 = 167.4 nM T40694 C7SR2D 52940661 IC50 = 35 nM T40694 CQVE12 52942317 IC50 = 200 nM T40694 CISC65 52943186 IC50 = 60 nM T40694 CKCN74 52943243 IC50 = 964 nM T40694 C2N5GH 52943310 IC50 = 8 nM T40694 C0LSU9 52944272 IC50 = 859 nM T40694 CE36VT 52944273 IC50 = 2650 nM T40694 C61JUX 52945276 IC50 > 10000 nM T40694 CF63AS 52945523 IC50 = 25 nM T40694 CQ30DI 52945929 IC50 = 33 nM T40694 CG8HT0 52946706 IC50 = 127 nM T40694 CQZX58 52946971 IC50 = 123 nM T40694 C84FOX 52946976 IC50 = 77 nM T40694 CRL93S 52947958 IC50 = 117 nM T40694 CP80TO 52947965 IC50 = 2682 nM T40694 C6O7CR 53249964 IC50 = 5.6 nM T40694 CFS57D 53261787 IC50 = 3290 nM T40694 C87LRX 53261846 IC50 = 1350 nM T40694 C25YMU 53261848 IC50 = 1260 nM T40694 CQW5Z9 53262909 IC50 > 20000 nM T40694 CIN3E9 53318794 IC50 < 9 nM T40694 C1CR6S 53363307 IC50 > 10000 nM T40694 CK03PA 53363389 IC50 > 10000 nM T40694 C8NA4L 53384644 IC50 > 30000 nM T40694 CU7SM4 53529356 IC50 > 10000 nM T40694 C30AQN 54580351 IC50 = 52 nM T40694 CEC0T9 54581348 IC50 = 154 nM T40694 CL42MV 54582373 IC50 = 6 nM T40694 CF7P8Y 54582374 IC50 = 279 nM T40694 C30RMF 54583357 IC50 = 42 nM T40694 CKM86O 54583358 IC50 = 201 nM T40694 CG9LS2 54583359 IC50 = 224 nM T40694 CY9J3B 54584304 IC50 = 44 nM T40694 CP2Z0T 54584305 IC50 = 83 nM T40694 CI4SU2 54585267 IC50 = 3 nM T40694 C51NCQ 54585268 IC50 = 60 nM T40694 CJ1S9E 54585269 IC50 = 106 nM T40694 CP86VM 54586220 IC50 = 43 nM T40694 C8WHP9 54587248 IC50 = 33 nM T40694 CFRA47 54675539 IC50 > 5000 nM T40694 CE1ZK6 54759168 IC50 = 15 nM T40694 C1XS2J 54760383 IC50 > 10000 nM T40694 C9ZFS1 54764923 IC50 > 100000 nM T40694 C8A4LW 55461102 IC50 = 1550 nM T40694 C6QGO9 56657855 IC50 = 15 nM T40694 CBZ8T4 56657856 IC50 = 6 nM T40694 CXIZ08 56659726 IC50 > 10000 nM T40694 CB3Q1P 56663194 IC50 > 10000 nM T40694 CA6T5S 56664839 IC50 = 6 nM T40694 CZYH57 56666592 IC50 > 10000 nM T40694 CYZ57N 56668250 IC50 = 4 nM T40694 CYPL60 56675140 IC50 = 4 nM T40694 C2BL7S 56676833 IC50 > 10000 nM T40694 CS3EP0 56676834 IC50 > 10000 nM T40694 CRG16Y 56676835 IC50 > 10000 nM T40694 C6B1PU 56676891 IC50 > 10000 nM T40694 CTBX87 56681780 IC50 = 7 nM T40694 CY36EG 56945171 EC50 = 64000 nM T40694 C4OG7H 56945172 EC50 = 440000 nM T40694 CH0QA3 56945173 IC50 = 10 nM T40694 CM0NQ5 56945174 IC50 = 7 nM T40694 CXKF03 56945175 IC50 = 4 nM T40694 CE07AQ 56945176 IC50 = 8 nM T40694 CY1U6R 56945271 EC50 = 150000 nM T40694 CU86KC 56945272 IC50 = 2 nM T40694 C9SX7F 56945273 IC50 = 1 nM T40694 CG7VH5 56945274 IC50 = 1 nM T40694 C62UBD 56945275 IC50 = 470 nM T40694 C6WU4V 56945277 EC50 = 44000 nM T40694 CH5Z0J 56946380 IC50 = 10 nM T40694 C4KS6O 56946480 IC50 = 18 nM T40694 CY4S5G 56946481 IC50 = 450 nM T40694 C81HTG 56946482 IC50 = 200 nM T40694 CP8VX7 56946483 IC50 = 65 nM T40694 CXS17A 56946484 IC50 = 83 nM T40694 CTS7U2 56946485 IC50 = 31 nM T40694 CL3YH1 56946582 IC50 = 120 nM T40694 C2ERQ5 56946583 IC50 = 78 nM T40694 C9Q0UX 56946584 IC50 = 33 nM T40694 C89OUI 56946585 IC50 = 370 nM T40694 CCH8B3 56946586 IC50 = 39 nM T40694 C91VNL 56946587 IC50 = 36 nM T40694 CBN5H2 56946588 IC50 = 120 nM T40694 CS28YK 56946691 IC50 = 340 nM T40694 C2NI9T 56946692 IC50 = 260 nM T40694 CVW45A 56946693 IC50 = 21 nM T40694 CQW0H1 56946694 EC50 = 630 nM T40694 C3JEI5 56946695 IC50 = 420 nM T40694 CY18FO 56946696 IC50 = 520 nM T40694 CZ1GF4 56946800 IC50 = 39 nM T40694 CMY32H 56946801 IC50 = 730 nM T40694 C8LOB3 56946803 IC50 = 130 nM T40694 CNSR78 56946804 IC50 = 290 nM T40694 CIV57W 56947168 IC50 = 820 nM T40694 CR16SD 56947170 IC50 = 5820 nM T40694 C84DVX 57386035 IC50 = 8410 nM T40694 CP68IC 57386289 IC50 = 3900 nM T40694 C16TMA 57386290 IC50 = 12100 nM T40694 C3R7OP 57386802 IC50 = 1320 nM T40694 CACW05 57386803 IC50 = 1560 nM T40694 C42HDB 57386804 IC50 = 3290 nM T40694 CNCO01 57386805 IC50 = 500 nM T40694 CG14VM 57387301 IC50 > 50000 nM T40694 CH53IA 57391401 IC50 = 3 nM T40694 CH53XJ 57391650 IC50 = 151 nM T40694 CF4U0R 57391651 IC50 = 817 nM T40694 CRLG52 57395119 IC50 = 272 nM T40694 CX6GJ7 57396885 IC50 = 102 nM T40694 CG4D3H 57398639 IC50 = 28 nM T40694 CMQ7A6 57400314 IC50 = 18 nM T40694 C3D6PW 57402024 IC50 = 130 nM T40694 C8H2MA 57402115 IC50 > 10000 nM T40694 CEG5Q7 57403865 IC50 = 18 nM T40694 CK7L8O 57403866 IC50 > 10000 nM T40694 CZSM95 57412684 IC50 > 10000 nM T40694 CUBP24 57955580 IC50 = 26 nM T40694 C0GKI6 57955606 IC50 = 190 nM T40694 CX4JP3 57955660 IC50 = 15 nM T40694 C73WGO 57955668 IC50 = 81 nM T40694 CG0C7J 57969945 IC50 = 70 nM T40694 CC7K8O 57970023 IC50 = 1 nM T40694 CL12XK 58009759 IC50 = 12 nM T40694 C4V7FY 58191950 IC50 = 27000 nM T40694 CPCA29 58191961 IC50 > 100000 nM T40694 C7HF1L 58191965 IC50 > 100000 nM T40694 C8LWY9 58191997 IC50 > 100000 nM T40694 CTV3K8 58405292 IC50 = 870 nM T40694 CNM93S 58405323 IC50 = 250 nM T40694 CCZ98N 58405467 IC50 = 250 nM T40694 CC90XE 58405504 IC50 = 1820 nM T40694 C29QLR 58405566 IC50 = 25300 nM T40694 C8RGV3 58405571 IC50 = 2340 nM T40694 CE69UL 58405593 IC50 = 3760 nM T40694 C2O3YU 58405631 IC50 = 8 nM T40694 C2L5SP 58405634 IC50 = 1820 nM T40694 C8QE2P 58405636 IC50 = 770 nM T40694 CE38BL 58405673 IC50 = 8670 nM T40694 CJG5F1 58405732 IC50 = 3420 nM T40694 CC8OS6 58405741 IC50 > 50000 nM T40694 CL7TF1 58405755 IC50 > 100000 nM T40694 CYN56J 58405790 IC50 = 1230 nM T40694 CDNU35 58405817 IC50 = 3550 nM T40694 C41DJO 58405910 IC50 = 9390 nM T40694 CDGV17 58405948 IC50 = 3030 nM T40694 CG63RM 58415665 IC50 = 7160 nM T40694 CXJ63M 59603829 IC50 > 100000 nM T40694 CQEU96 59603842 IC50 > 10000 nM T40694 COH62U 60097413 IC50 > 10000 nM T40694 C1MR8Q 60097495 IC50 > 10000 nM T40694 C4SGZ6 60165992 IC50 > 100000 nM T40694 C98NOD 60165993 IC50 = 60000 nM T40694 C3WIX5 60165994 IC50 > 100000 nM T40694 C0G5WC 60165995 IC50 > 100000 nM T40694 CEQ07N 60166135 IC50 > 100000 nM T40694 CRV13A 60166136 IC50 > 100000 nM T40694 CLP62H 60166137 IC50 = 15000 nM T40694 C9X0ZC 60166139 IC50 = 3700 nM T40694 CWPZ07 60166141 IC50 = 1200 nM T40694 CV63UL 67240318 IC50 > 10000 nM T40694 C8I7GC 68293638 IC50 > 10000 nM T40694 C2ZLY3 68310278 IC50 > 100000 nM T40694 C5DGR9 69036886 IC50 = 10000 nM T40694 C2HBG8 71450398 IC50 > 50 ug.mL-1 T40694 CMZ0V8 71450501 Ki = 14000 nM T40694 CY5P0T 71450502 Ki = 17600 nM T40694 C2PBG0 71450503 Ki = 14 nM T40694 CBQ6A4 71450504 Ki = 7720 nM T40694 CY38PM 71450505 Ki = 43 nM T40694 CPL36V 71450724 IC50 = 1100 nM T40694 C4CZ8D 71452343 Ki = 10 nM T40694 C62MTJ 71452344 Ki > 44000 nM T40694 CQYS65 71452345 Ki > 44000 nM T40694 CNV6K9 71452346 Ki = 315 nM T40694 C1EJ8I 71452347 Ki = 175 nM T40694 CEBO91 71452977 IC50 > 10000 nM T40694 C8AH1B 71454033 IC50 > 50 ug.mL-1 T40694 CI37UR 71454035 IC50 = 1.45 ug.mL-1 T40694 CX3AN8 71454037 IC50 > 50 ug.mL-1 T40694 CZ1V7O 71454128 Ki = 255 nM T40694 C4S9OQ 71454129 Ki = 1180 nM T40694 C1G0TW 71454130 Ki = 8530 nM T40694 CE5QY6 71454131 Ki = 13 nM T40694 CQL5Z9 71454309 IC50 = 170 nM T40694 CKT60L 71455860 Ki = 5 nM T40694 CCT9V1 71455861 Ki = 1800 nM T40694 CTSL27 71455862 Ki = 166 nM T40694 CGF6R1 71457661 Ki = 28 nM T40694 CTO38B 71457662 Ki = 1010 nM T40694 CO5IH0 71457663 Ki = 165 nM T40694 C7PZR2 71457664 Ki = 41 nM T40694 CADS56 71457665 Ki = 24900 nM T40694 CDYI16 71457666 Ki > 8800 nM T40694 CPNI86 71457857 IC50 = 320 nM T40694 C9ZVW4 71459442 IC50 = 7.54 ug.mL-1 T40694 CO9PR0 71459445 IC50 > 50 ug.mL-1 T40694 C8CO3A 71459558 Ki = 40800 nM T40694 CD0BG8 71459559 Ki = 75 nM T40694 C1JOZ2 71459560 Ki = 10 nM T40694 C89HGJ 71459561 Ki = 22 nM T40694 CD1OF0 71459769 IC50 = 140 nM T40694 CB9V6C 71461186 IC50 = 4.52 ug.mL-1 T40694 CF9K7H 71461301 Ki = 232 nM T40694 C0NZ4U 71461302 Ki = 47 nM T40694 C3B5WK 71461303 Ki = 4 nM T40694 CA3S8R 71461304 Ki = 15 nM T40694 CEB8I3 71461491 IC50 = 650 nM T40694 C6C4ZX 71461492 IC50 = 9300 nM T40694 CJ6T0K 71462927 IC50 = 6.87 ug.mL-1 T40694 CMV23P 71462929 IC50 = 10.06 ug.mL-1 T40694 CQG87Y 71463025 Ki = 20 nM T40694 CRU9F4 71463026 Ki = 82 nM T40694 CP4H5X 71463027 Ki = 85 nM T40694 C9ES8V 71463028 Ki = 333 nM T40694 CAU15Y 71463029 Ki = 276 nM T40694 CVM98J 71463030 Ki = 17 nM T40694 CJLX75 71468090 IC50 = 13000 nM T40694 CJQP29 71524012 IC50 = 139000 nM T40694 CCN01X 71547862 IC50 > 10000 nM T40694 CRX81Q 71575642 IC50 > 10000 nM T40694 CZ31PU 71583657 IC50 > 10000 nM T40694 C05ICM 71602777 IC50 = 320 nM T40694 CD7U3Q 71602778 IC50 = 380 nM T40694 C7BVZ4 71602779 IC50 = 480 nM T40694 CGOI91 71602780 IC50 = 7530 nM T40694 C64YHA 71602828 IC50 = 2830 nM T40694 C9B7LV 71602829 IC50 = 7760 nM T40694 CDSP70 71602874 IC50 = 28800 nM T40694 CUF0G5 71602875 IC50 = 3480 nM T40694 C9ZL1U 71602897 IC50 = 8500 nM T40694 CG58AU 71603001 IC50 = 2560 nM T40694 CB64UZ 71603062 IC50 = 1080 nM T40694 CO6I9D 71603063 IC50 = 4750 nM T40694 CLVQ91 71654873 IC50 = 1 nM T40694 CQ02SN 71664025 IC50 = 50 nM T40694 CJ4B7I 71682457 IC50 > 5000 nM T40694 CLI17Y 73351931 IC50 = 120 nM T40694 C7E2JD 73353563 IC50 = 1410 nM T40694 C8KH5E 73354910 IC50 = 9800 nM T40694 CE2Y0X 73386882 IC50 > 100000 nM T40694 C3UC9H 73891099 IC50 = 3180 nM T40694 CV8QX0 76310169 IC50 > 30000 nM T40694 CA5L4W 76324771 IC50 > 30000 nM T40694 C9GO0P 76328313 IC50 = 11800 nM T40694 C39FTZ 76335685 IC50 > 100000 nM T40694 CDG13U 86295201 Ki = 0.42 nM T40694 C1HW4B 89735655 IC50 > 100000 nM T40694 CFO48G 90643718 IC50 = 190 nM T40694 C07ZYI 90643719 IC50 = 30 nM T40694 CK49ZE 90643720 IC50 = 1550 nM T40694 CR1ZX5 90643721 IC50 = 590 nM T40694 CAV74K 90643722 IC50 = 1050 nM T40694 C6HPC3 90643723 IC50 = 190 nM T40694 C4W2UA 90643724 IC50 = 120 nM T40694 CYH3C7 90643725 IC50 = 90 nM T40694 C3AQ1G 90643726 IC50 = 2310 nM T40694 CY0UC4 90645194 IC50 > 10000 nM T40694 C0Y8ZK 91933875 IC50 > 1000 nM T40694 C0Q1FT 91938009 IC50 = 130 nM T40694 CGB54P 101902999 IC50 > 50000 nM T40694 CG62HP 101903000 IC50 > 50000 nM T40694 C4P7MG 118277818 Ki = 0.84 nM T40694 CKG9S0 118288047 Ki = 240 nM T40694 C8ZQL1 118288049 Ki = 0.91 nM T40694 CY7BI2 118706214 IC50 > 10000 nM T40694 C3KLI5 118723185 IC50 > 100000 nM T40694 C0QPN3 118726274 IC50 = 1820 nM T40694 C4O0EH 118726275 IC50 = 1910 nM T40694 C5A9BI 118726276 IC50 = 2100 nM T40694 CVGP61 118726277 IC50 = 4840 nM T40694 CV1E8I 118726278 IC50 = 3470 nM T40694 CRHT35 118726279 IC50 = 2640 nM T40694 C0KX2J 118726280 IC50 = 410 nM T40694 CL4VE6 118726281 IC50 = 1880 nM T40694 C3D0XF 118726282 IC50 = 960 nM T40694 CG3C9W 118726283 IC50 = 5710 nM T40694 CB9CT5 118726284 IC50 = 2900 nM T40694 CHT6K9 118728811 Ki > 4000 nM T40694 CUA3Y2 118728812 Ki > 4000 nM T40694 CDQ78G 118728813 Ki = 320 nM T40694 CZ6XL7 118728814 Ki = 1100 nM T40694 CMO67K 118728815 Ki = 1000 nM T40694 CR2M0Q 118728816 Ki > 4000 nM T40694 C62SCL 118728817 Ki > 4000 nM T40694 CSB30C 118728819 Ki = 2100 nM T40694 CV7XU8 118728820 Ki = 510 nM T40694 C3J1EX 118728821 Ki = 1700 nM T40694 CIWB78 118728822 Ki > 4000 nM T40694 CP18SE 118728823 Ki = 1000 nM T40694 CM42CA 118728824 Ki > 4000 nM T40694 C9Q7CL 118728825 Ki > 4000 nM T40694 CCR3S0 118728826 Ki > 4000 nM T40694 CD24VL 122187519 IC50 = 54.1 nM T40694 C8ZLB5 122187520 Ki = 4.2 nM T40694 C6OGU0 122187521 Ki = 6.95 nM T40694 CW84YE 122187522 Ki = 5.8 nM T40694 CH83IY 122187523 Ki = 0.52 nM T40694 C4X7SD 122192466 IC50 > 10000 nM T40694 C7GWV1 124098192 IC50 = 78 nM T40694 CQMU46 124201651 IC50 = 1.5 nM T40694 C2SO9N 134132792 IC50 = 164 nM T40694 C7DN4G 134137232 IC50 = 39800 nM T40694 CH9WC2 134139987 IC50 = 5050 nM T40694 CA2VM4 134140795 IC50 = 244 nM T40694 C8G0YI 134143573 IC50 = 91 nM T40694 CGI87V 134143656 IC50 = 119 nM T40694 C34EVY 134143682 IC50 = 6.6 nM T40694 CNW6Y3 134143807 IC50 = 94 nM T40694 CGM04X 134145100 IC50 = 43 nM T40694 C2H8KL 134146143 IC50 = 133 nM T40694 CK7P1W 134146150 IC50 = 163 nM T40694 CZ1N3R 134147429 IC50 = 149 nM T40694 CKN4T3 134148478 IC50 = 32 nM T40694 CAB06G 134148859 IC50 = 2380 nM T40694 CFB4E5 134150093 IC50 = 139 nM T40694 CS5ZU0 134151495 IC50 = 139 nM T40694 C1O6LZ 134152223 IC50 = 186 nM T40694 CHZD64 134157971 IC50 = 52 nM T40694 C2AN7T 134611886 IC50 > 100000 nM T40694 C2H7TQ 135473381 IC50 = 2000 nM T40694 CPV59N 135685787 Ki > 4000 nM T40694 C0CM9H 135879715 IC50 = 29000 nM T40694 C3YO9W 135929504 IC50 > 100000 nM T40694 C1NH5A 135929506 IC50 > 100000 nM T40694 CA8UN4 135929507 IC50 > 100000 nM T40694 C7J9ZD 135929508 IC50 > 100000 nM T40694 CB2P3H 135929509 IC50 > 100000 nM T40694 CJ1S7B 135929510 IC50 > 100000 nM T40694 C4IMU5 135929525 IC50 = 17000 nM T40694 C65NTO 135929526 IC50 > 100000 nM T40694 CAV34T 135929527 IC50 > 100000 nM T40694 C9EX0T 135929541 IC50 = 55000 nM T40694 CE4OU5 135929542 IC50 > 100000 nM T40694 C01HMT 135932346 IC50 > 10000 nM T40694 CF1PS8 135934877 Ki > 4000 nM T40694 CTRL59 135976660 Ki > 4000 nM T40694 C4RL7Q 135985508 IC50 > 10000 nM T40694 C8WIM5 135985510 IC50 > 10000 nM T40694 C3M7EP 135985511 IC50 = 24000 nM T40694 CMQ5W9 135985512 IC50 > 10000 nM T40694 CGM2H4 135988906 IC50 > 10000 nM T40694 CSO48W 135988918 IC50 = 49000 nM T40694 CXM18S 135988925 IC50 > 10000 nM T40694 C1ZT4N 135988927 IC50 > 10000 nM T40694 CVG5B9 135988940 IC50 = 15000 nM T40694 C68JXP 135988944 IC50 > 10000 nM T40694 CG23XF 135988947 IC50 > 10000 nM T40694 CIFX04 135988950 IC50 > 10000 nM T40694 CGP53C 135988956 IC50 = 26000 nM T40694 CLNJ17 135988957 IC50 > 10000 nM T40694 C7NU6A 135988961 IC50 > 10000 nM T40694 CR81AC 135988980 IC50 > 10000 nM T40694 C86BZJ 135988997 IC50 > 10000 nM T40694 C80PXZ 135989011 IC50 > 10000 nM T40694 CC6SO7 135989013 IC50 > 10000 nM T40694 CHA4N2 136013680 IC50 > 10 nM T40694 CQ84IZ 136180335 Ki > 4000 nM T40694 CZ7EX0 136183413 IC50 > 30000 nM T40694 C6HW4E 136206295 IC50 = 12000 nM T40694 CU9P3M 136206296 IC50 = 6000 nM T40694 C1YUD0 136219394 IC50 > 10 nM T40694 CY57SZ 136239319 IC50 = 10000 nM T40694 CJ2L3P 136239450 IC50 = 20000 nM T40694 C7XY0Q 136239451 IC50 = 15000 nM T40694 CN5LQ2 136239452 IC50 > 10000 nM T40694 CY08AS 136244133 IC50 > 10000 nM T40694 CIU8W3 136254389 IC50 > 10 nM T40694 C31BFH 137347775 IC50 = 290 nM T40694 C7FVC0 137347776 IC50 = 125 nM T40694 CH67OI 137631881 IC50 = 2.2 nM T40694 CH8YL3 137632392 IC50 = 9.7 nM T40694 C0XP4L 137632541 IC50 = 5.5 nM T40694 CG67CX 137633635 IC50 = 0.4 nM T40694 CE69HX 137637120 IC50 = 2 nM T40694 C72MFL 137640632 IC50 = 2.1 nM T40694 CXT65E 137642104 IC50 = 1.7 nM T40694 CFN5B9 137642203 IC50 = 8.6 nM T40694 C96RLN 137648227 IC50 = 45 nM T40694 C0UE7N 137648535 IC50 = 11.2 nM T40694 CV03IF 137648903 IC50 = 1.3 nM T40694 CN1LP0 137652774 IC50 = 5.5 nM T40694 C28QUP 137652864 IC50 > 10000 nM T40694 C7IH8L 137653047 IC50 = 7 nM T40694 C5E6CN 137653084 IC50 = 1.4 nM T40694 CY4JS5 137657338 IC50 = 1.9 nM T40694 C26LWI 137659622 IC50 = 2.2 nM T40694 CM3UF7 137700779 IC50 > 10000 nM T40694 CNP59S 141451364 IC50 = 33.1 nM T40694 C7QXC6 141451369 IC50 = 5.75 nM T40694 CM7O6D 141451370 IC50 = 38.02 nM T40694 CYHN75 141451372 IC50 = 16.05 nM T40694 CK1I8G 141451381 IC50 = 52.37 nM T40694 C6KQ8V 141451382 IC50 = 40.7 nM T40694 CRIZ46 141451383 IC50 = 34.94 nM T40694 C0QO5H 141451384 IC50 = 40.74 nM T40694 C78KWO 141451386 IC50 = 109 nM T40694 C09NZC 141451387 IC50 = 10.17 nM T40694 CJ21FB 145949301 IC50 = 2411 nM T40694 CA0RG8 145949395 IC50 = 1517 nM T40694 CCS05D 145950319 IC50 = 4991 nM T40694 C6LBJ2 145950482 IC50 = 121.5 nM T40694 C5L2IY 145950845 IC50 = 2556 nM T40694 CDT45G 145951146 IC50 = 62.25 nM T40694 CJ0H6I 145951269 IC50 = 97.75 nM T40694 C6J2FE 145951598 IC50 = 742 nM T40694 CWP5K3 145952451 IC50 = 5611 nM T40694 CAD7R9 145953240 IC50 = 4217 nM T40694 CEKL79 145954798 IC50 > 10000 nM T40694 CH0FJ8 145955296 IC50 = 460.1 nM T40694 CJ96ZH 145955626 IC50 = 882.7 nM T40694 C3TQ1E 145955731 IC50 = 64.77 nM T40694 C1AYV7 145957415 IC50 = 161.6 nM T40694 C5J7AZ 145957656 IC50 = 1147 nM T40694 C39VOT 145958071 IC50 = 3175 nM T40694 C9NPH7 145958192 IC50 = 284.2 nM T40694 CFGI54 145958286 IC50 = 93.79 nM T40694 C98TDA 145958548 IC50 = 1213 nM T40694 C1BJS3 145958954 IC50 = 1048 nM T40694 C2Z8NG 145960661 IC50 = 38.99 nM T40694 COK5G2 145960768 IC50 = 90.12 nM T40694 C5KRP1 145960780 IC50 = 79.84 nM T40694 CD3K7O 145961079 IC50 = 283.3 nM T40694 CNF8K3 145961137 IC50 = 75.27 nM T40694 CXD96P 145961248 IC50 = 74.14 nM T40694 CKJN89 145961654 IC50 = 46.58 nM T40694 C9OPQ4 145961681 IC50 = 65.59 nM T40694 C32IZF 145962002 IC50 = 70.24 nM T40694 C7TYS5 145962909 IC50 = 2109 nM T40694 CL56JT 145963032 IC50 = 78.42 nM T40694 C63ELA 145963541 IC50 = 2472 nM T40694 CC06PY 145963915 IC50 = 218 nM T40694 CDF9U4 145964106 IC50 > 12500 nM T40694 CC17DU 145964393 IC50 = 457 nM T40694 CH06LF 145964543 IC50 = 21 nM T40694 C87KPO 145964931 IC50 = 12350 nM T40694 CCW5X8 145965219 IC50 = 160 nM T40694 CN90GT 145965313 IC50 > 12500 nM T40694 CI9KC4 145965423 IC50 > 12500 nM T40694 CE4D5F 145966579 IC50 = 47 nM T40694 CXWZ04 145967512 IC50 = 25.2 nM T40694 CS6N3Y 145970287 IC50 = 2620 nM T40694 CQP70K 145971255 IC50 = 24.76 nM T40694 CIJO67 145972096 IC50 = 4 nM T40694 C0PFQ7 145972286 IC50 = 37.2 nM T40694 CN70KV 145972360 IC50 = 8.4 nM T40694 C2RTO8 145972845 IC50 = 8.7 nM T40694 CC8S9M 145972872 IC50 > 12500 nM T40694 CV4G1E 145973188 IC50 = 34.72 nM T40694 C7JIR5 145973809 IC50 = 43.41 nM T40694 C1HKY6 145973930 IC50 > 12500 nM T40694 CVU71O 145975475 IC50 = 673.5 nM T40694 C64XYG 145975479 IC50 = 461.6 nM T40694 CQA87Y 145975607 IC50 = 5910 nM T40694 C6SQL9 145975632 IC50 > 12500 nM T40694 C6R2YM 145975649 IC50 = 9.9 nM T40694 CTAZ41 145975701 IC50 = 322 nM T40694 CW56PH 145975703 IC50 = 40 nM T40694 CH57GW 145975937 IC50 = 4 nM T40694 CN4O0K 145976012 IC50 = 8.6 nM T40694 CR28YS 145976646 IC50 = 127 nM T40694 C5W8GH 145976701 IC50 > 12500 nM T40694 CCQS56 145977821 IC50 > 12500 nM T40694 CB9F1X 145977980 IC50 = 95 nM T40694 C0MD9U 145978238 IC50 = 27 nM T40694 C1MA9Q 145979724 IC50 = 6 nM T40694 C90QCO 145980261 IC50 = 5 nM T40694 CWL50V 145981755 IC50 = 85 nM T40694 CSY3K4 145987182 IC50 = 10 nM T40694 CY18PZ 145990069 IC50 = 370 nM T40694 CPY92M 155510533 IC50 = 68 nM T40694 C2MD1Q 155513187 IC50 > 10000 nM T40694 CQA75Z 155514946 IC50 = 5.14 nM T40694 CH82NV 155516034 IC50 = 26.77 nM T40694 C18XSD 155518015 IC50 = 3370 nM T40694 CQST37 155519017 IC50 = 10.17 nM T40694 CEI34U 155519091 IC50 = 5.76 nM T40694 CV40JF 155519344 IC50 = 6.86 nM T40694 CPS34K 155519748 IC50 = 540 nM T40694 C67ARO 155520726 IC50 = 123.8 nM T40694 C1SWX6 155520963 IC50 = 52.06 nM T40694 CUSF64 155521348 IC50 = 4.27 nM T40694 CLJ6B2 155522472 IC50 = 540 nM T40694 CTZ07V 155523554 IC50 = 884.6 nM T40694 CB2LE0 155524979 IC50 = 9.97 nM T40694 CQ0D4K 155525053 IC50 = 9.9 nM T40694 CLS4H2 155525411 IC50 = 84 nM T40694 C0P5XN 155525853 IC50 = 7.2 nM T40694 C4D3WX 155526889 IC50 = 3.89 nM T40694 CM1HB6 155527327 IC50 = 3.58 nM T40694 C9JT8G 155528462 IC50 = 20.72 nM T40694 C73EUH 155530844 IC50 = 7.28 nM T40694 CD65ZS 155533233 IC50 = 291.6 nM T40694 C1S6XO 155533569 IC50 = 110 nM T40694 CCL97M 155533912 IC50 = 177 nM T40694 CUI36R 155536170 IC50 = 126.3 nM T40694 CTSM92 155538441 IC50 = 8.8 nM T40694 CRWI29 155538752 IC50 = 1200 nM T40694 CM71YQ 155539415 IC50 = 17.29 nM T40694 CA9H6Y 155539913 IC50 = 126.8 nM T40694 CKR8W0 155541766 IC50 = 9.42 nM T40694 C69LPE 155543442 IC50 = 15.66 nM T40694 CMR1S9 155545273 IC50 = 17.9 nM T40694 CPUI60 155546408 IC50 = 400 nM T40694 CC1MU2 155546554 IC50 = 9.31 nM T40694 CB9V4S 155549112 IC50 = 5.89 nM T40694 C7R1IQ 155551215 IC50 = 52.61 nM T40694 CN5D6K 155552906 IC50 = 21.38 nM T40694 C6C1DL 155553924 IC50 = 21.21 nM T40694 CVQ5M8 155562100 IC50 = 2500 nM T40694 CSDM31 155562825 IC50 = 7.99 nM T40694 CU9HL1 155563487 IC50 = 20 nM T40694 C21DOA 155564098 IC50 = 30.31 nM T40694 CC1MR2 155566593 IC50 = 344.7 nM T40694 C4O8RS 155567235 IC50 = 1800 nM T40694 C3XS1Q 155568979 IC50 = 13.97 nM T40694 CR7LH1 9881974 Ki = 2000 nM T40694 D00ERW 44444843 Ki = 6560 nM T40694 D00HVA 11624601 Ki > 8900 nM T40694 D00JMT 210332 IC50 > 5000 nM T40694 D03DZO 11715767 IC50 = 980 nM T40694 D05QMQ 46235922 IC50 = 2 nM T40694 D05WDM 25015677 IC50 = 4 nM T40694 D06HVH 54613583 IC50 > 10000 nM T40694 D06QWO 14824655 IC50 > 10 ug.mL-1 T40694 D08HFG 24809764 IC50 > 10000 nM T40694 D09HVH 135566652 IC50 > 10 nM T40694 D09ZKY 25263088 IC50 = 9 nM T40694 D0A1CM 5281855 IC50 = 3340 nM T40694 D0D6MH 11617559 IC50 > 24000 nM T40694 D0F0AU 44405988 IC50 > 20000 nM T40694 D0G3SZ 6918469 IC50 = 7.1 ug.mL-1 T40694 D0J3LR 11634725 Ki > 4000 nM T40694 D0K0UJ 49837564 IC50 = 19400 nM T40694 D0L0HG 766949 IC50 > 10000 nM T40694 D0NJ4H 5281670 IC50 = 12600 nM T40694 D0Q3NG 11715520 Ki > 8900 nM T40694 D0QC0W 9914412 IC50 > 10000 nM T40694 D0S7IE 11658882 Ki > 8900 nM T40694 D0T8NU 16757525 IC50 = 574 nM T40694 D0UO2H 44556162 IC50 > 10000 nM T40694 D0X1RH 16051023 IC50 = 2 nM T40694 D0Z5TQ 5924208 IC50 = 4600 nM T42658 D0JU5X 400769 IC50 = 14080 nM T42658 C37TUW 122838 IC50 = 130 nM T42658 C2RG1J 2819993 EC50 = 4200 nM T42658 CK17XC 10422855 IC50 > 50000 nM T42658 CT0O5K 10634145 IC50 = 3800 nM T42658 CLT5R9 12019715 IC50 = 25000 nM T42658 CDQ6V8 16065919 IC50 = 420 nM T42658 CS24JL 17178045 IC50 > 2000000 nM T42658 C9C4TM 20866045 IC50 = 22600 nM T42658 CK7ZU4 20866046 IC50 = 28100 nM T42658 C3Z5CV 46830074 IC50 = 1600 nM T42658 C8W4MQ 46931952 IC50 = 6900 nM T42658 CIAN46 46931953 EC50 = 4200 nM T42658 CC6F2P 46931957 IC50 = 2200 nM T42658 CSX7K4 46932144 IC50 = 19000 nM T42658 CGOZ63 51031028 IC50 = 420 nM T42658 C8KW7D 54679359 IC50 = 2700 nM T42658 CK19RH 54691251 IC50 = 3500 nM T42658 CP5AM4 60207365 IC50 = 400 nM T42658 CJ6C9U 60207384 IC50 = 430 nM T42658 CLIX38 60207396 IC50 = 1700 nM T42658 CHQ3G4 60207417 IC50 = 380 nM T42658 CJ5RX4 60207506 IC50 = 7800 nM T42658 CT1MP7 67494944 IC50 = 380 nM T42658 CQU30L 68758187 EC50 = 20100 nM T42658 CQO45S 71278897 IC50 = 15000 nM T42658 CCTL58 71453283 IC50 > 31600 nM T42658 CT42XD 73345951 IC50 = 22600 nM T42658 C4F9RS 73349008 IC50 = 28000 nM T42658 CEU7P1 86276129 IC50 > 100000 nM T42658 CPC50V 90479863 IC50 > 50000 nM T42658 C94MHN 90479865 IC50 > 50000 nM T42658 CRW16J 102339098 IC50 = 490 nM T42658 CHE4A1 118352313 IC50 = 22570 nM T42658 CDJA36 118352321 IC50 = 3650 nM T42658 CJK51T 118352324 IC50 = 1350 nM T42658 CWE2V8 118352333 IC50 > 50000 nM T42658 CO5G1B 118352334 IC50 > 50000 nM T42658 CIL63V 118352335 IC50 = 4490 nM T42658 CWQ86Z 118352339 IC50 = 2650 nM T42658 C43SRU 118352342 IC50 = 6950 nM T42658 CQJD38 118352355 IC50 > 50000 nM T42658 CJQ5X2 118352358 IC50 = 26780 nM T42658 CZEJ62 118352364 IC50 = 670 nM T42658 CYD34F 118352365 IC50 > 50000 nM T42658 C59MPE 118352366 IC50 = 9930 nM T42658 C5IV6R 118352367 IC50 = 18020 nM T42658 CTI64U 118352368 IC50 = 4490 nM T42658 CUD4L7 118352369 IC50 = 16750 nM T42658 C4EFL9 118352370 IC50 > 50000 nM T42658 CNK75B 118352376 IC50 = 6120 nM T42658 C1A3ST 118352379 IC50 = 4210 nM T42658 CD5CH3 118352380 IC50 = 40490 nM T42658 C2NDW3 121435237 IC50 < 200 nM T42658 CZB39I 122531706 IC50 = 7600 nM T42658 C61RZG 122531715 IC50 = 5200 nM T42658 CD3YG9 122531725 IC50 = 13600 nM T42658 CTN05R 122531737 IC50 = 2500 nM T42658 C2IE5C 122531745 IC50 = 2500 nM T42658 CCO01X 122531747 IC50 = 610 nM T42658 CI93YD 122531750 IC50 = 1340 nM T42658 C2X7EH 122531784 IC50 = 480 nM T42658 CET68J 122531786 EC50 = 300 nM T42658 CMRF83 122531790 EC50 > 50000 nM T42658 CY95SO 122531794 IC50 = 21400 nM T42658 C8FWK4 122531796 IC50 = 9600 nM T42658 CZ7J4H 122531801 IC50 = 22400 nM T42658 C08LCX 126559338 IC50 = 130 nM T42658 CK51MI 126559339 IC50 = 75 nM T42658 CATC10 126559346 IC50 = 100 nM T42658 CYT9G6 126672795 IC50 = 15100 nM T42658 C9FW0X 131750078 IC50 = 6 nM T42658 CDZ28K 131750081 IC50 = 300 nM T42658 C9O2QW 131750084 IC50 = 46000 nM T42658 C3QM9R 131750085 IC50 = 13000 nM T42658 CAI2D1 131750087 IC50 = 300 nM T42658 CQAR36 131750088 IC50 = 22 nM T42658 C53HKL 131750089 IC50 = 2400 nM T42658 C70XSR 131953451 IC50 = 90 nM T42658 C47OID 132990905 IC50 = 90 nM T42658 CP25ZW 134451155 IC50 = 560 nM T42658 CSBJ35 134451172 IC50 = 90 nM T42658 C02HEJ 134451180 IC50 = 30 nM T42658 CR9W7E 134451182 IC50 = 39 nM T42658 CHU38F 134451185 IC50 = 40 nM T42658 CD4JO2 134451202 IC50 = 1900 nM T42658 CXZO30 134451210 IC50 = 120 nM T42658 C07LCS 134451218 IC50 = 240 nM T42658 C2FS5D 134451245 IC50 = 7200 nM T42658 CC4UW9 134451266 IC50 = 30 nM T42658 CWNX07 134451274 IC50 = 300 nM T42658 C1K4VE 134451275 IC50 = 44000 nM T42658 C8OCR9 134451347 IC50 = 130000 nM T42658 CN8BP5 134451350 IC50 = 115000 nM T42658 C2GL3U 134451359 IC50 = 150 nM T42658 CA2B9V 134451372 IC50 = 1400 nM T42658 CGF3R8 134451392 IC50 = 23000 nM T42658 C4GT9P 134451400 IC50 = 250 nM T42658 CAJO10 134451418 IC50 = 2800 nM T42658 C16IQU 134451421 IC50 = 87000 nM T42658 CUA52P 134451444 IC50 = 390 nM T42658 CO40LJ 134451448 IC50 = 35 nM T42658 CBO21N 134451450 IC50 = 24 nM T42658 CM8ZS6 134451452 IC50 = 330 nM T42658 CTM60B 134451499 IC50 = 90000 nM T42658 C58BUD 135567363 IC50 = 79200 nM T42658 C0GOR7 136699782 IC50 = 132000 nM T42658 CD43PS 137002862 IC50 = 97700 nM T42658 C2D7YU 137637373 IC50 = 85200 nM T42658 C9H6SI 137637597 IC50 = 8500 nM T42658 C9NR5M 137645854 IC50 > 200000 nM T42658 CP7N5G 137649194 IC50 = 131000 nM T42658 CSKX31 137650818 IC50 = 18400 nM T42658 CNK72M 137653175 IC50 = 33200 nM T42658 CLN32V 137659816 IC50 = 11100 nM T42658 CSC5I4 137659969 IC50 = 32800 nM T42658 C50YEW 138512896 IC50 = 4200 nM T42658 CZ5B0F 139414732 IC50 = 12000 nM T42658 CH8P5U 139414769 IC50 = 20000 nM T42658 C96WCT 139414836 IC50 = 50 nM T42658 CCOM78 145952644 IC50 < 200 nM T42658 C1ALP2 145961029 IC50 = 750 nM T42658 C4JXC5 145961432 IC50 = 200 nM T42658 CLOD21 145961463 IC50 = 8200 nM T42658 C6SM1N 145961517 IC50 < 500 nM T42658 C2S9EI 145961661 IC50 = 170 nM T42658 CB4K7Y 145962161 IC50 = 200 nM T42658 C7EDI0 145962970 IC50 = 300 nM T42658 CV71AX 145963074 IC50 = 200 nM T42658 CR2B7S 145963452 IC50 = 2000 nM T42658 CT38LW 145972867 IC50 = 2800 nM T42658 C2N0RF 145978273 IC50 = 4600 nM T42658 CR2DI7 145980365 IC50 = 8000 nM T42658 CR78YE 145981076 IC50 = 32000 nM T42658 CW3K6D 145982483 IC50 = 34000 nM T42658 CEW08J 145984129 IC50 > 200000 nM T42658 C63CMR 145988528 IC50 = 1400 nM T42658 CVTM05 145989351 IC50 = 23000 nM T42658 CWR39Y 145991193 IC50 = 10000 nM T42658 CQN12Y 145992545 IC50 = 78000 nM T42658 CJ2I4Q 145993154 IC50 = 60000 nM T42658 CQ2FK3 145993357 IC50 = 1100 nM T42658 CV9O0R 145993507 IC50 = 75 nM T42658 C5AW9L 146013528 IC50 = 44000 nM T42658 C0TE7M 155539687 IC50 = 52 nM T42658 CN7O1J 155568046 IC50 = 1.5 nM T42658 D07LUJ 64945 IC50 = 7000 nM T42658 D0I9UP 16065773 IC50 = 420 nM T69091 D01BYB 5957 EC50 = 56 nM T69091 D06JGH 1051 IC50 = 10000 nM T69091 D0UF2N 21706 EC50 = 182 nM T69091 CCJ8P0 440317 EC50 = 2300 nM T69091 CIWV85 746996 IC50 = 20700 nM T69091 CMUV80 766793 IC50 = 25200 nM T69091 CEBX03 779113 IC50 = 68800 nM T69091 CGJ9S2 921624 IC50 = 69600 nM T69091 CYV85L 2320735 IC50 >= 10000 nM T69091 CJEV94 5287422 EC50 = 6 nM T69091 C6P7VU 5311303 EC50 = 1150 nM T69091 CX92YW 6093160 IC50 = 210 nM T69091 CX7J8F 11636756 IC50 = 63.1 nM T69091 CR8U0Y 11663667 IC50 = 3000 nM T69091 CZF70G 24883277 IC50 > 10000 nM T69091 CQ46IG 44353592 EC50 = 2 nM T69091 CBPD97 46175179 IC50 > 10000 nM T69091 C80DAS 46231312 IC50 > 10000 nM T69091 C2W8ID 46832336 IC50 > 10000 nM T69091 CR98BF 53350233 IC50 = 1600 nM T69091 C8Z5FQ 60150614 IC50 = 180 nM T69091 CO7PZ5 60168729 IC50 = 6520 nM T69091 CH9Q0R 71450180 IC50 > 10000 nM T69091 CR64QG 71457337 IC50 > 10000 nM T69091 CR1L5W 71459185 IC50 = 602 nM T69091 CSV43Z 71459189 IC50 = 2020 nM T69091 C0Y1JN 71462707 IC50 >= 10000 nM T69091 CRZ62F 73355036 IC50 = 4270 nM T69091 C3U1YM 73669299 IC50 = 5320 nM T69091 CB69EX 76324694 IC50 = 4550 nM T69091 CPO7N5 124125214 IC50 > 50000 nM T69091 CLS0X7 145960885 IC50 > 10000 nM T69091 CF6LV4 155514310 IC50 > 100000 nM T69091 CM9CW2 155526224 IC50 > 100000 nM T69091 C1NOD4 155529242 IC50 = 41100 nM T69091 CX12AU 155529713 IC50 >= 10000 nM T69091 C5BC9V 155529971 IC50 > 100000 nM T69091 COD7Q8 155543044 IC50 = 8060 nM T69091 CZ9G8K 155559078 IC50 > 100000 nM T69091 C0PYX1 155562454 IC50 > 10000 nM T69091 D00QLM 91557 EC50 = 200 nM T69091 D05NWF 6022 EC50 = 10000 nM T69091 D0B1KT 15953802 IC50 > 10000 nM T69091 D0U1OJ 5310983 EC50 = 54 nM T69091 D0UG4S 91532 EC50 = 2000 nM T69091 D0V4GQ 5310996 EC50 = 2500 nM T71907 CBLH67 3236077 EC50 = 9900 nM T71907 C3FCP6 3240071 EC50 = 860 nM T71907 C0W2VJ 6619083 EC50 = 1400 nM T71907 CINB06 17253251 EC50 = 8800 nM T71907 CWU3Z8 17253286 EC50 = 1800 nM T71907 CSVT87 17253337 EC50 = 1500 nM T71907 CJW1E2 53016936 EC50 = 280 nM T71907 C2YW1K 53016939 EC50 = 260 nM T71907 C7L2NR 53016945 EC50 = 2800 nM T71907 C28EIO 72710837 EC50 = 290 nM T71907 C37HBK 73051406 EC50 = 3560 nM T71907 CC43AX 73051560 EC50 = 1930 nM T71907 CC73KY 73051561 EC50 = 5500 nM T71907 CBRM50 89932298 EC50 = 260 nM T71907 CX83DO 110856568 EC50 = 5400 nM T71907 CM3Q8S 110856660 EC50 = 1800 nM T71907 CT4DI5 110856964 EC50 = 720 nM T71907 C46DVJ 110858626 EC50 = 1800 nM T71907 CK0N9O 110858729 EC50 = 6200 nM T71907 CA2EZ7 110859813 EC50 = 7300 nM T71907 CMY51K 110859918 EC50 = 3600 nM T71907 C5ODV2 110862668 EC50 = 340 nM T71907 CSEJ78 137631523 EC50 = 13900 nM T71907 CN79TO 137635641 EC50 = 780 nM T71907 CF0VK6 137639244 EC50 = 500 nM T71907 CWZ9L4 137643290 EC50 = 1600 nM T71907 CFC3V5 137643971 EC50 = 9900 nM T71907 CN3L2O 137644369 EC50 = 11200 nM T71907 CY14WM 137646891 EC50 = 2600 nM T71907 CV73IM 137647050 EC50 = 360 nM T71907 C1EVG0 137652995 EC50 = 500 nM T71907 CO90YW 137655778 EC50 = 170 nM T36612 CFB4W1 253688 IC50 = 170 nM T36612 C1HYD5 265935 IC50 = 4400 nM T36612 C7KQ3Z 11589584 Ki = 293000 nM T36612 C0U7YP 13891339 IC50 = 710 nM T36612 CTE72N 51049631 IC50 = 390 nM T36612 C1MFN2 54756939 IC50 = 34000 nM T36612 COF2G6 54756941 IC50 = 690 nM T36612 CH69FL 146680924 IC50 = 5400 nM T36612 C54VSY 155515570 IC50 = 19000 nM T36612 C1VN8A 155520618 IC50 = 7300 nM T36612 C7CU2H 155528540 IC50 = 12000 nM T36612 CH5VR7 155530421 IC50 = 5800 nM T36612 C6VO9W 155536240 IC50 = 5600 nM T36612 CDY59I 155553395 IC50 = 10700 nM T36612 CZR6D8 155553413 IC50 = 65000 nM T36612 D01FNC 21771691 IC50 = 130 nM T36612 D02ZNQ 5298 IC50 = 430 nM T36612 D0YP0A 24970878 IC50 = 6000 nM T07191 D0OB0F 5328940 IC50 = 9.9 nM T07191 D03BNU 59604787 IC50 > 10000 nM T07191 CUJR40 10062694 IC50 = 28 nM T07191 CE36DN 11156201 IC50 = 42 nM T07191 CJ5W9L 11181283 IC50 = 8 nM T07191 C3TOH4 11191242 IC50 = 33 nM T07191 C0YH2X 11478363 IC50 = 8 nM T07191 CZV0O2 12003241 IC50 = 5 nM T07191 C5VPH9 16129448 IC50 = 115 nM T07191 CCP2M3 24822704 IC50 > 50000 nM T07191 CC71QJ 27666048 IC50 > 100000 nM T07191 CLW80F 44160269 IC50 = 2600 nM T07191 CK73NR 44219749 IC50 > 50000 nM T07191 C4WRN5 44541014 IC50 = 50000 nM T07191 C3VRO9 44557921 IC50 > 10000 nM T07191 C28QLM 44605035 IC50 > 50000 nM T07191 C75XHS 44605037 IC50 > 50000 nM T07191 CC95PQ 45375865 IC50 = 1300 nM T07191 CEOQ27 45375866 IC50 > 50000 nM T07191 C96BNW 46179972 IC50 = 24 nM T07191 CO3P0J 46866604 IC50 < 50000 nM T07191 CLS29B 46872626 IC50 > 10000 nM T07191 CJOM49 46880136 IC50 = 4100 nM T07191 CWM9H3 46900076 IC50 = 47 nM T07191 CR8T3P 59711970 IC50 = 925 nM T07191 COH62U 60097413 IC50 > 5000 nM T07191 C1MR8Q 60097495 IC50 > 2500 nM T07191 C37NKO 67129970 IC50 = 4760 nM T07191 CK80LJ 67130050 IC50 = 6240 nM T07191 CV63UL 67240318 IC50 > 10000 nM T07191 C7GRV2 68755406 IC50 = 1570 nM T07191 CDJY72 71568837 IC50 = 3000 nM T07191 C8CAG7 71578921 IC50 > 10000 nM T07191 CQ53SW 71682214 IC50 = 9700 nM T07191 C5N1VZ 102581295 IC50 > 10000 nM T07191 CM3WO6 134304664 IC50 = 7 nM T07191 CR6L0B 134304723 IC50 = 6 nM T07191 C2AN7T 134611886 IC50 > 100000 nM T07191 CGBZ13 134843302 IC50 = 1200 nM T07191 C3MK9W 136807986 IC50 > 10000 nM T07191 CXC69T 137321158 IC50 = 387 nM T07191 CXP53D 137348835 IC50 = 1 nM T07191 CI1E8V 137634241 IC50 = 2940 nM T07191 C49KUQ 145964145 IC50 = 24 nM T07191 CE5S1W 145964374 IC50 = 27 nM T07191 CPVG78 145964598 IC50 = 10 nM T07191 C9MX1N 145964844 IC50 = 39 nM T07191 CP83FM 145964889 IC50 = 63 nM T07191 CL3H4Z 145965408 IC50 = 1080 nM T07191 CSK06W 145966254 IC50 = 14 nM T07191 CWK7C2 145966484 IC50 = 17 nM T07191 C6RXU9 145967106 IC50 = 497 nM T07191 CK0CV9 145970783 IC50 = 45 nM T07191 C0Y2WF 145972806 IC50 = 55 nM T07191 CAGL67 145972836 IC50 = 16 nM T07191 C4J5YX 145976700 IC50 = 8 nM T07191 CF6NW2 145976762 IC50 = 34 nM T07191 C5RX9K 145977177 IC50 = 5 nM T07191 CJE14S 145977878 IC50 = 72 nM T07191 CJ07WY 145978202 IC50 = 2 nM T07191 C75UKW 145978330 IC50 = 165 nM T07191 CN58FM 145978369 IC50 = 2 nM T07191 C68GMW 155538446 IC50 > 10000 nM T07191 CY6Q8S 155554337 IC50 = 40000 nM T07191 CO2I4P 155559898 IC50 = 600 nM T07191 D00ERW 44444843 Ki > 6516 nM T07191 D05MHL 44605611 Ki = 340 nM T07191 D09PTP 57325421 IC50 = 60 nM T50089 D07UHS 107970 EC50 = 0.3 nM T50089 D07EDB 52938427 EC50 = 4.3 nM T50089 D07FKQ 44599207 EC50 = 0.98 nM T50089 D07UGA 5283560 EC50 = 0.2 nM T50089 D0I2RB 11502996 EC50 = 0.33 nM T50089 D0L9KH 44623998 EC50 = 24.4 nM T50089 D0K4BI 10223146 IC50 > 1000 nM T50089 D0PW0R 71547555 IC50 > 10000 nM T50089 C3RZ6P 904918 EC50 > 10000 nM T50089 C7QC0W 1776080 EC50 = 721 nM T50089 CPO6B9 2740144 IC50 > 10000 nM T50089 C7N5UR 4107292 IC50 > 10000 nM T50089 CIA43B 4492589 IC50 = 14000 nM T50089 CS8MB9 9821227 EC50 > 5000 nM T50089 CW37CN 9969355 EC50 = 170 nM T50089 C7FGR9 9979368 IC50 = 0.8 nM T50089 CI3K9Z 10023913 EC50 = 41 nM T50089 CZLT30 10045980 IC50 = 1 nM T50089 CN8H2S 10127475 IC50 = 23 nM T50089 CCG97S 10127776 IC50 = 10 nM T50089 C5XFN7 10174255 IC50 = 16 nM T50089 C5HJB9 10195325 IC50 = 120 nM T50089 C6NP8S 10217498 IC50 = 18 nM T50089 CN93ZD 10249887 IC50 = 5.2 nM T50089 C6H9VI 10249979 IC50 = 12 nM T50089 C2O4UR 10251062 IC50 = 11 nM T50089 C5MDF6 10288527 IC50 = 13 nM T50089 CPK61C 10310952 IC50 = 77 nM T50089 C3SM5Z 10317453 IC50 = 1.6 nM T50089 CG89DO 10363915 IC50 = 1.8 nM T50089 C8WL6R 10408874 IC50 = 0.5 nM T50089 COQ65E 10409838 IC50 = 6.4 nM T50089 CI3EW1 10430549 IC50 = 1 nM T50089 CAL72D 10476387 IC50 = 6.6 nM T50089 C9NRD6 11168252 IC50 = 21 nM T50089 CZ3T0G 11177439 EC50 = 2400 nM T50089 CD8T1W 11222939 EC50 = 0.46 nM T50089 CUR1P8 11224984 EC50 = 59.1 nM T50089 CFPH94 11248292 IC50 = 41 nM T50089 CK65MP 11271470 IC50 = 10 nM T50089 CYH0U8 11408903 IC50 = 12 nM T50089 CER35T 11466640 IC50 = 53 nM T50089 CW51YT 11495139 IC50 = 300 nM T50089 CDE78J 11496072 EC50 = 3.9 nM T50089 C7EOU1 11501764 IC50 = 48 nM T50089 CR1ME9 11501873 EC50 = 530 nM T50089 CS27OX 11502026 IC50 = 1000 nM T50089 CL50IH 11503967 IC50 = 1360 nM T50089 CAG0Y9 11540052 IC50 = 122 nM T50089 C3BK8V 11568622 EC50 = 0.92 nM T50089 CVW6Q3 11575787 IC50 = 0.4 nM T50089 CB75ZP 11575913 EC50 = 43 nM T50089 CXS54Q 11603220 IC50 = 12 nM T50089 C5BDY3 11603528 EC50 = 150 nM T50089 CCW90K 11603726 EC50 = 73 nM T50089 C96LNP 11604577 IC50 = 0.5 nM T50089 CAN4Q9 11611053 EC50 = 820 nM T50089 C7I6ZU 11619303 EC50 = 0.98 nM T50089 C41XAE 11624780 EC50 > 1000 nM T50089 CCY7J2 11626664 EC50 = 24 nM T50089 C4IMA6 11632823 EC50 = 220 nM T50089 CA8W5N 11646599 EC50 = 210 nM T50089 CYS5F1 11653967 IC50 = 4 nM T50089 C8TL6P 11654374 EC50 = 120 nM T50089 CMJ32O 11662328 EC50 = 9.9 nM T50089 CQTW52 11675496 EC50 > 10000 nM T50089 C8CQ2N 11675907 EC50 = 26 nM T50089 CD4AO7 11676168 EC50 = 21 nM T50089 CCNU48 11678855 EC50 = 1.995 nM T50089 C3Q9JR 11682677 EC50 = 12 nM T50089 CVG41H 11682696 EC50 = 270 nM T50089 CQRA36 11683935 IC50 = 104 nM T50089 CCF80W 11689680 EC50 = 6.5 nM T50089 C8XLO4 11690779 IC50 = 455 nM T50089 C0BR1U 11696807 IC50 = 20 nM T50089 CK5S1L 11697013 EC50 = 950 nM T50089 C4G2OP 11743459 IC50 = 0.3 nM T50089 CZ6YN9 11752659 IC50 = 33 nM T50089 CLHA36 11869937 EC50 = 1760 nM T50089 C03OUS 11977938 EC50 = 17 nM T50089 CDI32A 16038017 EC50 = 44 nM T50089 CGAD08 17253208 EC50 > 25000 nM T50089 C0O9UG 24825338 EC50 = 40 nM T50089 CB82GW 24825339 EC50 = 28.6 nM T50089 C1TGE9 25008420 IC50 = 9.6 nM T50089 C1EM2P 25154344 EC50 = 114 nM T50089 C6RM3T 25182621 EC50 = 258 nM T50089 CP1CA9 25182769 EC50 = 191 nM T50089 CF35EH 25182773 EC50 = 96 nM T50089 CGEM35 25182899 EC50 = 142 nM T50089 CNYW93 25182926 EC50 = 6.3 nM T50089 C10HKX 25192001 EC50 = 0.33 nM T50089 C48TPJ 42630194 EC50 = 11 nM T50089 CDL1C8 44125170 EC50 = 162.18 nM T50089 CG73ST 44138103 EC50 = 21 nM T50089 C95GIJ 44342175 EC50 = 52 nM T50089 C7YT1J 44342219 EC50 = 43 nM T50089 C8NOT7 44342221 EC50 = 645.5 nM T50089 CCN68O 44342231 EC50 = 1220 nM T50089 CXJ08Y 44342244 EC50 = 1606 nM T50089 C6LT8S 44342246 EC50 > 5000 nM T50089 CLXY90 44342331 EC50 = 160 nM T50089 CI01UD 44342339 EC50 = 55 nM T50089 CAUQ90 44342468 EC50 = 110 nM T50089 CJ36UD 44394116 IC50 = 24 nM T50089 C5KA6D 44394117 IC50 = 680 nM T50089 CU7L0K 44394153 IC50 = 34 nM T50089 CT8UN6 44394161 IC50 = 230 nM T50089 C9E6CF 44394169 IC50 = 660 nM T50089 C8H0XM 44394191 IC50 = 0.58 nM T50089 CH2A5S 44394211 IC50 = 270 nM T50089 CND39O 44394212 IC50 = 61 nM T50089 C84JPI 44394247 IC50 > 1000 nM T50089 CA28OJ 44394273 IC50 = 1.2 nM T50089 CO0T1E 44394279 IC50 = 17 nM T50089 CE25XJ 44394289 EC50 = 370 nM T50089 C0X4ZS 44394327 EC50 = 77 nM T50089 CL5BC6 44394330 IC50 > 1000 nM T50089 CU3KA2 44394460 EC50 = 8.2 nM T50089 C24XDE 44394498 EC50 = 6.6 nM T50089 CZ14XU 44394521 EC50 = 390 nM T50089 C6XO8W 44394564 EC50 = 2400 nM T50089 CI75GS 44398012 EC50 = 51 nM T50089 CCFT02 44398049 EC50 = 16 nM T50089 CRYM50 44398058 EC50 = 37 nM T50089 CR3K9W 44398074 EC50 = 6700 nM T50089 C4DIT3 44398076 EC50 = 17 nM T50089 C3H2IY 44398170 EC50 = 29 nM T50089 CL5SY3 44398172 EC50 = 860 nM T50089 CR4TH0 44406004 EC50 = 1.995 nM T50089 C3JF1Q 44406009 EC50 = 50.12 nM T50089 CDY46P 44412165 IC50 = 13 nM T50089 CR2DT4 44412221 IC50 = 1280 nM T50089 CRV34X 44412232 IC50 = 180 nM T50089 CV63YC 44412233 IC50 = 200 nM T50089 CQ1V3J 44412282 IC50 = 100 nM T50089 CB6KR7 44412294 IC50 = 30 nM T50089 CTV5M0 44412353 IC50 = 30 nM T50089 CN7K2O 44412364 IC50 = 16 nM T50089 CL1GJ3 44412415 IC50 = 80 nM T50089 CV28IK 44412416 IC50 = 20 nM T50089 CBM50W 44412428 IC50 = 60 nM T50089 C2US0I 44412578 EC50 = 43 nM T50089 CM46YR 44412604 EC50 = 3200 nM T50089 C1LTZ6 44412605 EC50 = 3200 nM T50089 C28CAY 44412621 EC50 = 460 nM T50089 C9I7UV 44412622 EC50 > 10000 nM T50089 CNF3Y2 44412623 EC50 > 10000 nM T50089 CG7T1N 44412643 EC50 > 10000 nM T50089 C05TUB 44412658 EC50 > 10000 nM T50089 CH51GD 44412659 EC50 > 10000 nM T50089 C93OLQ 44412660 EC50 > 10000 nM T50089 C0CA6R 44412661 EC50 = 200 nM T50089 CL54DN 44412674 EC50 > 10000 nM T50089 C3M5SO 44412702 EC50 > 1000 nM T50089 CBUQ92 44412827 EC50 = 1080 nM T50089 CM8IK4 44412854 EC50 = 4000 nM T50089 C34QEC 44412865 EC50 = 1300 nM T50089 CBL87K 44412867 EC50 = 260 nM T50089 COA6Q1 44412868 EC50 = 2600 nM T50089 C80JSN 44412882 EC50 = 591 nM T50089 C2WV6S 44412883 EC50 = 840 nM T50089 C84PLZ 44412908 EC50 = 266 nM T50089 C78DOK 44412936 EC50 = 15 nM T50089 CH6Z8V 44412962 EC50 > 10000 nM T50089 C3MWD4 44412971 EC50 = 3.1 nM T50089 CJC06H 44412994 EC50 = 0.7 nM T50089 CT6EU7 44413274 IC50 = 130 nM T50089 CYO6R3 44413349 IC50 = 5.1 nM T50089 CH9NL4 44413365 IC50 = 21 nM T50089 CW8E0R 44413415 IC50 = 390 nM T50089 CYW5D3 44413430 IC50 = 140 nM T50089 CJ5S2H 44413446 IC50 = 68 nM T50089 CWRZ40 44413447 IC50 = 57 nM T50089 CVC61G 44413482 IC50 = 50 nM T50089 CWL92R 44422573 EC50 = 76 nM T50089 C12CHR 44422579 EC50 = 41 nM T50089 C0I3LB 44422601 EC50 = 30 nM T50089 C2O7AP 44422604 EC50 = 19 nM T50089 C07YCS 44422605 EC50 = 31 nM T50089 C7O0PC 44422606 EC50 = 47 nM T50089 C0W3FQ 44439850 EC50 = 5.1 nM T50089 CB4Z3I 44439851 EC50 = 5.2 nM T50089 C9SFT8 44439852 EC50 = 37.7 nM T50089 CS9H0L 44517795 EC50 = 109 nM T50089 CX13MK 44547414 EC50 = 88 nM T50089 CP18DA 44565596 IC50 = 43.6 nM T50089 CO8AD3 44565597 IC50 = 2.9 nM T50089 CS13TE 44565622 IC50 = 26.2 nM T50089 COH39N 44565714 IC50 = 70.4 nM T50089 CB1GT5 44565715 IC50 = 99.8 nM T50089 CAV3F9 44565716 IC50 = 207 nM T50089 C76DFZ 44565717 IC50 = 9.6 nM T50089 CMG7L1 44565738 IC50 = 12.8 nM T50089 CH8SJ9 44565739 IC50 = 3.5 nM T50089 CX9AZ4 44591249 IC50 = 8.8 nM T50089 C3NOY0 44591250 IC50 = 6.9 nM T50089 C3TAY6 44591264 IC50 = 3.2 nM T50089 CGCL62 44591265 IC50 = 1.4 nM T50089 C10TGI 44591266 IC50 = 1.1 nM T50089 C1GW4T 44600476 EC50 = 29 nM T50089 C6T4QB 45377662 EC50 = 62 nM T50089 C73DCB 46174905 EC50 = 81 nM T50089 CSTA18 46224712 EC50 = 900 nM T50089 C4QB8F 46224713 EC50 > 10000 nM T50089 C4HN6L 46224714 EC50 = 325 nM T50089 CF75RO 46224715 EC50 = 82 nM T50089 C6R9SJ 46224716 EC50 > 10000 nM T50089 CB56OX 46224767 EC50 = 130 nM T50089 CHC1D9 46224768 EC50 = 345 nM T50089 C15WRO 46224769 EC50 = 505 nM T50089 CMW59H 46225233 EC50 > 10000 nM T50089 CV5T1F 46225282 EC50 > 10000 nM T50089 CF74HE 46225283 EC50 > 10000 nM T50089 C6XAU7 46225284 EC50 > 10000 nM T50089 CL4H8B 46225285 EC50 > 10000 nM T50089 CQY5P8 46866185 EC50 = 200 nM T50089 C6LJ7A 46866186 EC50 = 280 nM T50089 CD2HV5 46872048 IC50 = 9 nM T50089 CFM69E 46872386 IC50 = 277 nM T50089 CJN7K1 46872388 IC50 = 13 nM T50089 CS62XM 46872389 IC50 = 7 nM T50089 CP0A4M 46872507 IC50 = 255 nM T50089 C13OBR 46872619 IC50 = 1 nM T50089 CB8IG2 46872620 IC50 = 5 nM T50089 CL69YZ 46872622 IC50 = 6 nM T50089 CTM7O9 46872625 IC50 = 789 nM T50089 CLS29B 46872626 EC50 = 4.1 nM T50089 CZ7PU2 46872748 IC50 = 1210 nM T50089 C04MNL 46872872 IC50 = 28 nM T50089 C6HL5D 46872874 IC50 = 16 nM T50089 CQZ59G 46881623 EC50 = 0.6 nM T50089 CW6RX2 46881847 EC50 = 2.2 nM T50089 CAHC81 46881875 EC50 = 19 nM T50089 CCS12Z 46881877 EC50 = 3600 nM T50089 C3QMS1 46881912 EC50 = 1000 nM T50089 CTL89X 46884020 EC50 = 1.49 nM T50089 CJ21TY 46885796 IC50 = 87.2 nM T50089 CZDL71 46885798 IC50 = 184 nM T50089 CG9X7Z 49830722 IC50 = 1 nM T50089 CS6JN0 49830723 IC50 = 2 nM T50089 CJ3CQ5 49830724 IC50 = 2 nM T50089 CS1NI2 49830725 IC50 = 4 nM T50089 C84YOW 49830828 IC50 = 4 nM T50089 C3SAE6 49830919 IC50 = 1 nM T50089 CCX14T 49835928 EC50 = 2100 nM T50089 CS25XW 49835989 EC50 = 237 nM T50089 C5Z6RM 49839234 EC50 = 5.8 nM T50089 C4BXP1 49848557 EC50 = 16.6 nM T50089 CMV6Y2 49868651 EC50 = 0.53 nM T50089 CH0B8K 50925337 EC50 = 1.1 nM T50089 C1DYT0 53358422 IC50 = 5500 nM T50089 CC7DZ4 53362086 EC50 = 19 nM T50089 CG3FA9 53492750 EC50 = 19.95 nM T50089 C5M2PI 54580603 IC50 > 20000 nM T50089 CWNO65 54582607 IC50 = 3000 nM T50089 CU62DN 54764919 EC50 = 4300 nM T50089 C1RK0O 57390238 EC50 = 3400 nM T50089 CKWG20 57390239 EC50 = 144 nM T50089 CT9J5U 57390243 EC50 = 196 nM T50089 CM74JH 57395471 EC50 = 6180 nM T50089 CPY57D 57397320 EC50 = 51 nM T50089 C3KS0A 57397321 EC50 = 22 nM T50089 CT7E0J 57398996 EC50 = 652 nM T50089 CXO9I1 57398998 EC50 = 37 nM T50089 CS3I9U 57400714 EC50 = 34 nM T50089 CLG2V4 57554674 IC50 < 1 nM T50089 COE91B 57699087 Ki > 10000 nM T50089 C5YS7U 58329611 EC50 > 10000 nM T50089 C8FZ4S 59384310 EC50 = 0.66 nM T50089 CQ52OA 59384375 EC50 = 2 nM T50089 CDA7S4 59451739 IC50 = 35 nM T50089 CV3RJ6 59451743 IC50 = 115 nM T50089 CE47JS 59451750 IC50 = 8 nM T50089 C0SP8Q 59451751 IC50 = 125 nM T50089 C3D4EZ 59451753 IC50 = 7 nM T50089 C1CYE5 59451764 IC50 = 9 nM T50089 CF5VO8 59451770 IC50 = 10 nM T50089 CC81PQ 59451779 IC50 = 26 nM T50089 CQ7J3Z 59451780 IC50 = 75 nM T50089 C7L4SK 59451793 IC50 = 1 nM T50089 C3Q9PE 59451795 IC50 = 32 nM T50089 CC9FN3 59451797 IC50 = 23 nM T50089 CG1YS4 59451808 IC50 = 5 nM T50089 CQ23ZL 59451812 IC50 = 10 nM T50089 CU83BX 59451813 IC50 = 3 nM T50089 CLQ46R 59451819 IC50 = 2 nM T50089 C7CR6Z 59451824 IC50 = 409 nM T50089 CB9S0P 59451832 IC50 = 77 nM T50089 CRE85M 59451845 IC50 = 5 nM T50089 C0KJ1F 59451849 IC50 = 5 nM T50089 CK3IM1 59451852 IC50 = 8 nM T50089 CIR58O 59451857 IC50 = 8 nM T50089 CV94QR 59451859 IC50 = 41 nM T50089 CR62AY 59451867 IC50 = 148 nM T50089 CCAI45 59451870 IC50 = 3 nM T50089 CR8NC6 59451874 IC50 = 2 nM T50089 CVY6T4 59451878 IC50 = 108 nM T50089 CVN69I 59451883 IC50 = 16 nM T50089 C7YA0P 66655198 EC50 = 15.85 nM T50089 CMT3L8 66655210 EC50 = 12.59 nM T50089 C1M4BX 66655282 EC50 = 63.1 nM T50089 CD09QP 66655362 EC50 = 19.95 nM T50089 CD2I5L 66655520 EC50 = 125.89 nM T50089 CTX2M1 66655578 EC50 = 31.62 nM T50089 CASW54 66655584 EC50 = 31.62 nM T50089 CN83CO 66655586 EC50 = 199.53 nM T50089 CJG3A2 66655632 EC50 = 25.12 nM T50089 CI5KQ1 66655655 EC50 = 12.59 nM T50089 CSVZ95 66655679 EC50 = 15.85 nM T50089 CRGW91 66655753 EC50 = 199.53 nM T50089 C9PGA0 66655774 EC50 = 6.31 nM T50089 C7WVE9 66655956 EC50 = 158.49 nM T50089 CZS20N 66655962 EC50 = 100 nM T50089 C6UGD4 66655998 EC50 = 39.81 nM T50089 CQ0U7L 66656025 EC50 = 316.23 nM T50089 CKO1L6 66656274 EC50 = 1000 nM T50089 C5UTG1 66829311 EC50 = 753 nM T50089 C6AZY0 67249162 EC50 = 410 nM T50089 CX6SF2 67250226 EC50 = 47 nM T50089 CR2TI7 68489165 IC50 = 9 nM T50089 CY09OV 69263869 EC50 = 275 nM T50089 CR4V0T 71450073 IC50 = 978 nM T50089 C9IKU5 78321974 EC50 = 10.7 nM T50089 CI1WF3 89710483 EC50 = 125.89 nM T50089 C2G1HE 89710485 EC50 = 25.12 nM T50089 CJ6RC9 89710536 EC50 = 1995.26 nM T50089 CGE95T 89710694 EC50 = 7.943 nM T50089 CLP73T 89710808 EC50 = 63.1 nM T50089 CR0LX1 89711073 EC50 = 19.95 nM T50089 C2D4SQ 89713031 EC50 = 2.512 nM T50089 C0TQK5 89713056 EC50 = 15.85 nM T50089 CL74JM 90309142 IC50 > 10000 nM T50089 C72NCP 118728432 IC50 > 10000 nM T50089 CH23UV 124171442 EC50 = 350 nM T50089 C9VT4Z 124171444 EC50 = 340 nM T50089 CX8VT2 124171447 EC50 = 360 nM T50089 CONE63 124171453 EC50 = 215 nM T50089 C9U4QR 124221654 EC50 = 370 nM T50089 CQ37LX 127037695 IC50 = 1 nM T50089 CM54QV 127037696 IC50 = 9 nM T50089 CD52GS 127041987 IC50 = 5 nM T50089 C01YZA 134129958 EC50 = 1070 nM T50089 C9XCH3 134129983 EC50 = 412 nM T50089 CVYH81 134130022 EC50 = 2590 nM T50089 COK2V9 134130023 EC50 = 728 nM T50089 CK3D4G 134130066 EC50 = 49 nM T50089 C9J4YQ 134130071 EC50 > 100000 nM T50089 CO7NQ6 134130111 EC50 = 272 nM T50089 CDFI08 134130114 EC50 = 2320 nM T50089 C2XC8U 134130131 EC50 = 10260 nM T50089 CAOF06 134130145 EC50 > 100000 nM T50089 CCMS20 134130146 EC50 = 4220 nM T50089 C4KI5E 134130150 EC50 = 329 nM T50089 CUE0N7 134130169 EC50 = 22 nM T50089 CNW53I 134130183 EC50 = 4510 nM T50089 CVA1C4 134130188 EC50 = 2490 nM T50089 CS0W9B 134130192 EC50 = 887 nM T50089 C90GZS 134130203 EC50 > 100000 nM T50089 CYS41M 134130243 EC50 > 100000 nM T50089 C25EHG 134130292 EC50 > 100000 nM T50089 CHXD46 134130316 EC50 = 350 nM T50089 C7K1UH 134130375 EC50 = 2810 nM T50089 C4B2LQ 134130519 EC50 = 25 nM T50089 CE3O4Z 134130538 EC50 = 21200 nM T50089 C3NC1O 134130546 EC50 = 31 nM T50089 CJH4K9 134130548 EC50 = 356 nM T50089 CD9YI4 134130571 EC50 = 1670 nM T50089 C3YO7L 134130622 EC50 > 100000 nM T50089 CD7W9Y 134130662 EC50 = 232 nM T50089 C6JB4Z 134130695 EC50 = 51 nM T50089 CMX5L2 134130704 EC50 > 100000 nM T50089 CE9AV5 134130732 EC50 = 3070 nM T50089 C6V4DA 134130884 EC50 = 152 nM T50089 CGK8F7 134130947 EC50 = 6450 nM T50089 C4FBV1 134130960 EC50 > 100000 nM T50089 CFU7G1 134131038 EC50 > 100000 nM T50089 CP67CL 134131039 EC50 > 100000 nM T50089 CXKZ69 134131043 EC50 = 6700 nM T50089 CU93MF 134131067 EC50 = 4020 nM T50089 CV20CR 134131071 EC50 = 143 nM T50089 C1F7MJ 134131075 EC50 > 100000 nM T50089 C2VW9K 134131081 EC50 = 280 nM T50089 CJBU52 134131130 EC50 > 100000 nM T50089 CJI9U7 134131169 EC50 = 4690 nM T50089 CLM0H7 134131188 EC50 = 1560 nM T50089 CA86SG 134131209 EC50 = 3970 nM T50089 CX84LY 134131253 EC50 > 100000 nM T50089 C2OEB6 134131256 EC50 = 3130 nM T50089 C6GE4C 134131291 EC50 = 506 nM T50089 CBKF68 134131297 EC50 = 709 nM T50089 C2SJ7C 134131301 EC50 = 2140 nM T50089 CCH9O4 134131316 EC50 = 769 nM T50089 CFR58S 134131363 EC50 = 552 nM T50089 CNVC46 134131381 EC50 = 60 nM T50089 CE13OT 134131399 EC50 = 3540 nM T50089 CS13QG 134131470 EC50 = 2100 nM T50089 C9UB6W 134131475 EC50 = 4770 nM T50089 C64QZX 134131495 EC50 > 100000 nM T50089 C09ZOI 134131497 EC50 > 100000 nM T50089 C6DJ2N 134131598 EC50 = 175 nM T50089 CH2AN7 137660780 IC50 > 10000 nM T50089 CHRG61 145964044 EC50 = 794.33 nM T50089 C0ZM4R 145966230 IC50 > 1000 nM T50089 CR8Q4L 145969830 EC50 = 316.23 nM T50089 CN8IE0 145975394 EC50 = 15.85 nM T50089 C6JW8K 145976329 IC50 > 1000 nM T50089 C7MI9V 145978086 EC50 = 19.95 nM T50089 CRF7V0 155317229 IC50 > 1000 nM T50089 CX76PB 155317261 IC50 > 1000 nM T50089 CW10AC 155317265 IC50 > 1000 nM T50089 C43CXP 155317276 IC50 > 1000 nM T50089 CLG86C 155317279 IC50 > 1000 nM T50089 CPY85W 16215109 EC50 = 10.2 nM T50089 CZSI05 44438257 EC50 = 133.8 nM T50089 CWKU57 44438259 EC50 = 5.8 nM T50089 CT3AX1 44438261 EC50 = 21.3 nM T50089 D00VHN 46905530 IC50 = 0.77 nM T50089 D02LTS 59393720 IC50 > 10000 nM T50089 D04IAF 11452022 EC50 = 0.3 nM T50089 D05EDD 11588811 EC50 = 52 nM T50089 D05KEE 10904818 EC50 = 1.995 nM T50089 D06DYN 9908268 EC50 = 0.4 nM T50089 D06GFH 11545181 EC50 = 33 nM T50089 D06XMB 44394220 IC50 = 110 nM T50089 D07EAB 10215259 IC50 = 29 nM T50089 D0D5QS 11725751 IC50 = 8.2 nM T50089 D0LO4T 10287034 IC50 = 2.2 nM T50089 D0N0BN 44394248 IC50 > 1000 nM T50089 D0P1TY 44344193 IC50 = 13 nM T50089 D0P2AZ 10149721 IC50 = 11 nM T50089 D0ZU0O 4077460 IC50 = 4600 nM T15610 D0RA5Q 72172 IC50 = 3500 nM T15610 D0F2JS 15547703 IC50 = 260 nM T15610 CESM72 439530 IC50 = 2450 nM T15610 CV25HK 9900746 IC50 = 3800 nM T15610 CX98JA 10357930 IC50 = 3400 nM T15610 CEOM91 44381716 IC50 = 4600 nM T15610 CBKT65 44564374 IC50 = 1790 nM T15610 CU32WC 53348579 IC50 = 5000 nM T15610 C7A6QJ 73323710 IC50 = 68810 nM T15610 CYND40 90672013 IC50 = 940 nM T15610 CG9N2T 90672014 IC50 = 7.4 nM T15610 CMY4U5 127040069 IC50 = 8040 nM T15610 C95FOZ 127040083 IC50 = 36420 nM T15610 CTD3E7 127042345 IC50 = 92510 nM T15610 C0S7EH 127042346 IC50 = 80970 nM T15610 CJL98E 127042347 IC50 = 32680 nM T15610 CC82PR 127042676 IC50 = 8530 nM T15610 CEOW50 127042689 IC50 = 42960 nM T15610 CJ37ZH 127042690 IC50 = 92870 nM T15610 CQC5A9 127042691 IC50 = 36270 nM T15610 CP5R9K 127042981 IC50 = 98190 nM T15610 CGS9N5 127042982 IC50 = 10180 nM T15610 CLJ9F6 145949706 IC50 = 53000 nM T15610 CQNE67 145956257 IC50 > 100000 nM T15610 CBR41A 145957710 IC50 = 53000 nM T15610 CB03UD 145960195 IC50 = 4800 nM T15610 CZU0S1 145963748 IC50 = 1400 nM T15610 D0J0IY 44381715 IC50 = 2900 nM T20578 D0A9IY 135564558 IC50 > 10000 nM T20578 CX5HW2 376977 IC50 = 1500 nM T20578 CUK49V 11988837 Ki = 300 nM T20578 CFIO49 11988967 Ki = 910 nM T20578 C2D0NG 11989101 Ki = 1200 nM T20578 C65ABT 11989102 Ki = 6100 nM T20578 C1B4XD 11992634 IC50 > 2000 nM T20578 CPX16N 11993169 IC50 > 2000 nM T20578 C9WKV0 14531504 IC50 = 3000 nM T20578 CFAQ86 22343616 IC50 = 600 nM T20578 CW96SI 23624262 IC50 > 1000 nM T20578 C9WGI4 24802717 IC50 = 3100 nM T20578 C6EQG2 24963293 IC50 > 2000 nM T20578 C6R4YN 50993785 IC50 = 10000 nM T20578 C0M6XL 50993786 IC50 = 10000 nM T20578 CPC3T4 56654131 IC50 > 10000 nM T20578 CD52CA 57391118 IC50 > 2000 nM T20578 CY8J3O 68181896 IC50 = 12000 nM T20578 CC43LF 71074083 IC50 > 10000 nM T20578 CZ0G2X 72165213 IC50 > 10000 nM T20578 C7XRY6 72190879 IC50 > 30000 nM T20578 CQ3GD7 72704434 Ki = 360 nM T20578 C9JE6M 75815419 IC50 = 41.3 nM T20578 CQCA74 101886683 IC50 = 13900 nM T20578 C2L1SH 101886684 IC50 = 1410 nM T20578 COZ0H2 101886685 IC50 = 2200 nM T20578 CSCY01 117949009 IC50 > 10000 nM T20578 CRJE23 122185011 IC50 > 29800 nM T20578 C4UR7D 127038167 IC50 > 1000 nM T20578 C4H2TJ 127038168 IC50 > 1000 nM T20578 CL9JT8 127038169 IC50 > 1000 nM T20578 CJPX60 127038509 IC50 > 1000 nM T20578 C26EAG 127038511 IC50 > 1000 nM T20578 CTM9E4 127038512 IC50 > 1000 nM T20578 C6AQ2U 127038513 IC50 < 1000 nM T20578 CV1FM0 127038868 IC50 > 1000 nM T20578 CADU23 127038869 IC50 > 1000 nM T20578 C3R8SE 135457869 IC50 > 10000 nM T20578 CTX54Z 135896326 IC50 > 10000 nM T20578 C2FW0D 135981181 IC50 = 31 nM T20578 CJM3W6 135981182 IC50 = 8 nM T20578 C12UMG 136059728 IC50 > 1000 nM T20578 CE4HQ5 136230157 IC50 = 43 nM T20578 CH5SF7 136230158 IC50 = 11 nM T20578 CI1W8Q 136230159 IC50 = 19 nM T20578 C9Q2ZK 136254168 IC50 = 17 nM T20578 C2N9VT 137348687 IC50 > 10000 nM T20578 D06NIT 135564899 IC50 > 1000 nM T79027 D07XSN 6253 Ki = 190000 nM T79027 D0Y7DP 6029 Ki = 0.0012 nM T79027 D0I5OR 29243 Ki = 100 nM T79027 CJK3C5 94312 Ki = 40000 nM T79027 C5F6MJ 125382 Ki = 25100000 nM T79027 C1Q0KC 9543506 IC50 = 340 nM T79027 C67SRQ 9881381 IC50 = 13000 nM T79027 CVN49Q 21117530 Ki = 400 nM T79027 C84WEG 22677568 Ki = 1600000 nM T79027 C5CY4Q 25267009 IC50 = 400 nM T79027 C4FB8O 25267372 IC50 = 5000 nM T79027 C2MOV6 25267373 IC50 = 400 nM T79027 CH97QJ 25267374 IC50 = 5000 nM T79027 CGR4K5 25267375 IC50 = 200 nM T79027 CXG9J8 25267376 IC50 = 4000 nM T79027 C93YCO 44266514 Ki = 7690000 nM T79027 CK52DI 44320529 Ki = 100000 nM T79027 CI7PH4 46876305 Ki = 300000 nM T79027 CQ7N0R 46876306 Ki = 2800 nM T79027 CHA1N8 46876343 Ki = 25 nM T79027 C3S8RJ 46876842 Ki = 9000 nM T79027 CUX4T5 46876856 Ki = 15000 nM T79027 CK74TE 54227907 Ki = 40 nM T79027 CWKO70 57704491 IC50 = 20000 nM T79027 C3M8GN 57704511 IC50 > 100000 nM T79027 CU74CG 57704512 IC50 > 100000 nM T79027 C6DB3Z 57704515 IC50 = 77000 nM T79027 D0IF3H 100016 Ki = 2000 nM T06273 D01SHZ 9931954 IC50 = 0.8044 nM T06273 D04AIT 5280445 IC50 = 4265.8 nM T06273 D06NVJ 936 IC50 = 210000 nM T06273 D09LSX 11291932 IC50 = 7 nM T06273 D0GV8J 135565082 IC50 = 0.6 nM T06273 D0J9HW 23725625 Ki = 0.787 nM T06273 D00BMF 24958200 Ki = 3.2 nM T06273 D07OIO 44199317 IC50 = 1.7 nM T06273 D09NTC 9840076 Ki = 5.8 nM T06273 D0R2OU 25070031 IC50 > 30000 nM T06273 D09WUA 73669300 IC50 = 70 nM T06273 D0F5TD 135565981 IC50 = 2 nM T06273 D0E2VC 148140 Ki = 70 nM T06273 D0O3FX 135398517 Ki = 48 nM T06273 C6WGQ5 1340 IC50 = 390 nM T06273 CH62DB 1853 IC50 = 300 nM T06273 CD1Q4C 2331 IC50 = 20000 nM T06273 C8GAZ7 8394 IC50 = 12000 nM T06273 CGY7X0 8602 IC50 = 8500 nM T06273 CT4KV3 12084 IC50 = 300000 nM T06273 CH34LK 12576 IC50 = 160000 nM T06273 C7UQO3 65052 IC50 = 280000 nM T06273 C2TX3O 66491 IC50 = 1400 nM T06273 C6RV0E 68000 IC50 = 20000 nM T06273 CH1DK9 69253 IC50 = 19000 nM T06273 CN1G4Z 69254 IC50 = 22000 nM T06273 C1P6CX 69683 IC50 = 2200000 nM T06273 CX8O3Y 71572 IC50 = 200000 nM T06273 C9YN0B 76079 IC50 = 1800000 nM T06273 CXG7Y0 76959 IC50 = 57000 nM T06273 CY3VB9 89807 IC50 = 55000 nM T06273 CS74HZ 145726 IC50 = 1258.93 nM T06273 C7WS2Q 150896 IC50 = 100000 nM T06273 C2S0RK 157180 IC50 = 156 nM T06273 C3X0CZ 165356 IC50 = 900000 nM T06273 CL6K0E 206931 Ki = 105 nM T06273 C0F1IA 229015 IC50 = 2454.71 nM T06273 CJ2UB5 236501 IC50 > 100000 nM T06273 CY65EM 261391 IC50 = 10000 nM T06273 CN9Z6M 265048 IC50 = 240 nM T06273 CA6WM0 269082 IC50 = 312 nM T06273 CI80CO 269083 IC50 = 6100 nM T06273 C0CPI7 270668 IC50 = 180 nM T06273 CC82MK 276231 IC50 = 35000 nM T06273 C6TB1F 276271 IC50 = 180 nM T06273 CQ6OJ1 283716 IC50 = 3260 nM T06273 CA2C7O 354460 IC50 = 9570 nM T06273 C8S7VQ 360876 IC50 = 167 nM T06273 CMX2C1 448890 IC50 = 60 nM T06273 CWB45K 482198 IC50 = 22000 nM T06273 CDY93O 576186 Ki = 45 nM T06273 CYC75Z 622510 IC50 = 2600 nM T06273 C1XBG2 659976 IC50 = 4100 nM T06273 C8AW6J 676438 IC50 = 4200000 nM T06273 CAH3Q5 687511 IC50 = 1920 nM T06273 CQ21MC 717725 IC50 = 3600 nM T06273 CJA32Z 722008 IC50 = 724.44 nM T06273 C5X1HK 823807 IC50 = 1660 nM T06273 CSOZ61 1157122 IC50 = 720 nM T06273 CSW76H 1556947 IC50 = 1960 nM T06273 CZG84L 1577619 IC50 = 2140 nM T06273 C37IQB 2058875 IC50 = 4400 nM T06273 C5B0WQ 2106442 IC50 > 20000 nM T06273 C3DJT0 2393489 IC50 = 2100 nM T06273 C7Y6UE 2474690 IC50 = 42.9 nM T06273 CQ6WD1 2740936 Ki = 238 nM T06273 C2R7PJ 2758498 IC50 = 120000 nM T06273 C89WXS 2802462 IC50 = 19100 nM T06273 CB0N7J 2821781 IC50 > 25000 nM T06273 CK24BY 3014425 IC50 = 500000 nM T06273 C9PKJ8 3041095 Ki = 47 nM T06273 CX6KD5 3238600 IC50 = 1140 nM T06273 CV21AQ 3796800 IC50 = 97 nM T06273 CR26SK 4163640 IC50 > 100000 nM T06273 C5QTJ0 4438821 IC50 = 2010 nM T06273 CT9V6M 4826644 IC50 > 100000 nM T06273 C4QO1U 4849074 IC50 = 690 nM T06273 C7M9XJ 5309879 Ki = 172 nM T06273 C4C8BV 5320693 IC50 > 100000 nM T06273 CB86MY 5391140 IC50 = 9500 nM T06273 C7CIL3 6490174 IC50 > 100000 nM T06273 CW9FY1 6918639 IC50 > 1000000 nM T06273 C4P2UQ 8607850 IC50 > 100000 nM T06273 CB6QU2 9794892 Ki < 5 nM T06273 CH9YG2 9795674 Ki = 11 nM T06273 C0B6IA 9795692 Ki = 11 nM T06273 CWEY13 9796149 IC50 = 45 nM T06273 CF2C4S 9814168 IC50 = 800 nM T06273 CF28MZ 9814194 IC50 = 111 nM T06273 C5IMN8 9815456 Ki = 38 nM T06273 CQ4B7F 9817572 EC50 = 15 nM T06273 C7Z4HT 9817600 Ki = 4.5 nM T06273 CW7Q6I 9839073 IC50 = 68 nM T06273 CJ45OI 9839168 Ki = 11 nM T06273 CQVL57 9857216 IC50 = 26 nM T06273 CH75GJ 9861308 Ki < 5 nM T06273 CUF3C6 9861852 Ki = 8 nM T06273 CQ40VY 9864119 IC50 = 14 nM T06273 C37IGA 9868833 IC50 = 20 nM T06273 CDQF05 9878580 IC50 = 37 nM T06273 CB9NE2 9879829 Ki = 4.9 nM T06273 C3LSI2 9882962 Ki = 3.8 nM T06273 C9ZG4K 9884838 IC50 = 20 nM T06273 CI5O3Y 9889396 EC50 = 10 nM T06273 CAV3P4 9899130 IC50 = 900 nM T06273 CPBU63 9903811 Ki = 5 nM T06273 C6CHD2 9904310 Ki = 5.7 nM T06273 C9WJ5O 9904988 IC50 = 12 nM T06273 CED20G 9905158 Ki = 6.3 nM T06273 CNX6F7 9921542 Ki = 5 nM T06273 CD2K3N 9921681 IC50 = 36 nM T06273 CEZ80X 9922091 IC50 = 44 nM T06273 CP02XQ 9922953 IC50 = 118 nM T06273 C4IH1C 9924905 IC50 = 25 nM T06273 CVN86P 9925900 Ki = 59 nM T06273 CFND51 9943191 Ki = 4.1 nM T06273 CK1P9J 9943215 IC50 = 700 nM T06273 C6H4RC 9944838 IC50 = 17 nM T06273 CEF9Q5 9945164 IC50 = 162 nM T06273 CXA70E 9948137 Ki = 8 nM T06273 CYT5D3 9948349 IC50 = 53.2 nM T06273 C91UMH 9967081 IC50 = 59 nM T06273 CY9V5R 9970889 Ki < 5 nM T06273 CL97WP 9993998 IC50 = 30 nM T06273 CNYT58 10002219 EC50 = 300 nM T06273 C5OUY2 10039306 Ki = 3.2 nM T06273 C07YSN 10081381 IC50 = 2600 nM T06273 CRV4E7 10085156 Ki = 8 nM T06273 C6W4TV 10085758 IC50 = 10 nM T06273 CK48UD 10105388 EC50 > 3000 nM T06273 CD7IP9 10111909 IC50 = 25 nM T06273 CZM3R2 10117105 IC50 = 20 nM T06273 CLGZ29 10130109 Ki = 95 nM T06273 CJ12OG 10132635 IC50 = 35 nM T06273 C7S6DE 10134062 IC50 = 376 nM T06273 C2VTF7 10135674 IC50 = 20 nM T06273 C2U6AE 10135782 IC50 = 13 nM T06273 C5H6KM 10150882 IC50 = 119 nM T06273 CAG19D 10155051 IC50 = 457 nM T06273 C01TYD 10155422 IC50 = 150 nM T06273 C2PJD3 10157622 IC50 = 13 nM T06273 CJYG60 10158853 IC50 = 16 nM T06273 C1ZE4L 10159521 IC50 = 32 nM T06273 C5Z3MV 10177097 IC50 = 33 nM T06273 CW5GL2 10194337 IC50 = 16 nM T06273 C58RQB 10200345 IC50 = 21 nM T06273 C20STJ 10216071 IC50 = 46 nM T06273 C7EHI5 10220882 Ki = 6 nM T06273 CD6X1R 10221158 Ki = 44 nM T06273 CTI8Z3 10224010 IC50 = 30 nM T06273 C5GK4Z 10230030 IC50 = 20 nM T06273 CH6B2R 10237099 IC50 = 64 nM T06273 C94TAV 10241296 Ki = 99 nM T06273 CS25YP 10242492 IC50 = 20 nM T06273 C3F8CN 10267996 IC50 = 88 nM T06273 CA6YN5 10292240 IC50 = 63 nM T06273 CP5JZ9 10297291 IC50 = 357 nM T06273 C1R8UY 10366554 IC50 = 25 nM T06273 C95MLS 10375426 IC50 = 169 nM T06273 C0VN9K 10423087 Ki = 6.8 nM T06273 CD6N3Y 10424118 IC50 = 29 nM T06273 C3F0QA 10450266 Ki = 1.4 nM T06273 C2N5DC 10466183 IC50 = 270 nM T06273 CMQ9L2 10472074 IC50 = 71 nM T06273 CACP56 10492366 Ki = 9.4 nM T06273 CPN52M 10540758 Ki = 5.9 nM T06273 CN5UH4 10540772 Ki = 32 nM T06273 COC8G7 10585483 Ki = 350 nM T06273 CXK54M 10587888 Ki = 6.8 nM T06273 C2RGL0 10598394 Ki = 85 nM T06273 CQ8OB4 10615886 Ki = 9.4 nM T06273 CNE9A1 10634624 Ki = 6.3 nM T06273 CK8BU1 10659747 Ki = 3 nM T06273 C4LX8M 10683256 Ki = 10.6 nM T06273 C4R1WA 10684365 Ki = 2 nM T06273 CX80KN 10707280 Ki = 8.4 nM T06273 CYWZ68 10710001 Ki = 8.1 nM T06273 CIX47D 10729476 Ki = 11 nM T06273 C2IVK4 10730177 Ki = 4 nM T06273 C8EGS0 10755250 Ki = 290 nM T06273 CR3M1J 10758576 Ki = 136 nM T06273 CP2H7W 10778228 Ki = 1.6 nM T06273 CW1GJ8 10801775 Ki = 126 nM T06273 C4LXZ5 10804503 Ki = 1.2 nM T06273 C1TO3E 10823781 Ki = 15 nM T06273 CWSJ85 10824891 Ki = 9 nM T06273 CAU3M2 10827834 Ki = 5.4 nM T06273 CD87EP 10828391 Ki = 190 nM T06273 C2T4EO 10834881 Ki = 530 nM T06273 CFU9A5 10850356 Ki = 5.8 nM T06273 C2A9BW 10852098 Ki = 8 nM T06273 CP3SE1 10867239 IC50 = 14000 nM T06273 C4SZ5H 10867569 IC50 = 209 nM T06273 C0XJD4 10871043 IC50 = 339 nM T06273 C8J2ZW 10878066 IC50 = 2900 nM T06273 C4LVH3 10881392 Ki = 32 nM T06273 CL9DG7 10891646 Ki = 6 nM T06273 COHX01 10928352 IC50 = 142 nM T06273 C03SJB 10935844 IC50 = 865.3 nM T06273 C6FW5B 10936513 IC50 = 98 nM T06273 CWD09N 10938033 IC50 = 774 nM T06273 CN0S7L 10944628 Ki = 14 nM T06273 CZB5N6 10956768 Ki = 7 nM T06273 COF08D 10970760 IC50 = 111 nM T06273 C2IX4R 10970843 IC50 = 58 nM T06273 C1FGU3 10971050 IC50 = 75 nM T06273 C8SLD1 10979819 IC50 = 247 nM T06273 CTB73Z 10980119 Ki = 5 nM T06273 C5CEU9 10990023 Ki = 4.2 nM T06273 CVCK13 10991133 Ki = 6 nM T06273 C3OV7I 10999499 Ki = 8 nM T06273 C2VXJ6 11010927 Ki > 10000 nM T06273 CQ1D6S 11012595 Ki = 29 nM T06273 CT7IE1 11012966 Ki = 11.2 nM T06273 CN4U8B 11014815 Ki = 230 nM T06273 C4WQT7 11015219 IC50 = 86 nM T06273 CT1V2L 11044477 Ki > 10000 nM T06273 C4W3UX 11044567 Ki = 8.8 nM T06273 C0AMD4 11044955 Ki < 5 nM T06273 CPVF53 11054997 Ki = 23 nM T06273 CZUI30 11067571 IC50 = 165 nM T06273 CWG0N3 11078020 Ki = 5 nM T06273 CXT48V 11091010 IC50 = 277 nM T06273 CSO1X6 11109746 Ki = 5 nM T06273 CF1H0T 11129411 Ki = 32 nM T06273 CW90OL 11130277 Ki = 7.7 nM T06273 C2VI9R 11138393 Ki = 11 nM T06273 CJ5DH1 11161961 IC50 > 10000 nM T06273 C3AI6C 11162143 Ki = 8.2 nM T06273 CY79GV 11186827 Ki = 219 nM T06273 C65HZN 11186992 Ki = 79 nM T06273 CRAT13 11195895 Ki = 809 nM T06273 CVN57Z 11202184 EC50 = 70 nM T06273 CR1MQ0 11229916 Ki = 606 nM T06273 C0HZP7 11230287 Ki = 900 nM T06273 CGV6H0 11231597 Ki = 27 nM T06273 C2P3XT 11232005 Ki = 6.9 nM T06273 CQ0ND6 11248095 EC50 = 9 nM T06273 CUM91H 11252639 Ki = 122 nM T06273 CY1M7X 11257357 EC50 = 400 nM T06273 C6BEU4 11269254 IC50 > 3000 nM T06273 CQZC62 11289389 Ki = 22 nM T06273 C8X9OG 11290531 EC50 = 650 nM T06273 C6R8GB 11298843 Ki = 176 nM T06273 COI8C4 11300812 Ki = 380 nM T06273 CPO7X9 11301623 Ki = 9.1 nM T06273 CLDZ24 11301786 Ki = 43 nM T06273 CH0Y7I 11311554 Ki = 14.3 nM T06273 C8PMG5 11324750 Ki = 200 nM T06273 C7LAY1 11335260 Ki = 337 nM T06273 CP2IH0 11336230 Ki = 306 nM T06273 CIX6H4 11336543 EC50 = 80 nM T06273 CPO7C3 11336928 Ki = 249 nM T06273 C9XV5U 11338625 EC50 = 9 nM T06273 CC26LQ 11378922 Ki = 79 nM T06273 CUMO64 11381183 Ki = 54 nM T06273 C0HAQ1 11392596 EC50 = 65 nM T06273 CHJ3E5 11393561 Ki = 9.1 nM T06273 CW15FY 11403138 Ki = 41 nM T06273 C4W9ZQ 11408838 EC50 = 300 nM T06273 CLG82H 11436466 Ki = 121 nM T06273 C3NE4R 11439016 EC50 = 28 nM T06273 C2SIC4 11448426 Ki = 68 nM T06273 C80XTJ 11464583 IC50 > 3000 nM T06273 CZ39MJ 11483768 Ki = 304 nM T06273 C65MLE 11553859 IC50 = 188 nM T06273 C8LK1S 11670314 IC50 = 36 nM T06273 CF2I6K 11675005 IC50 = 4.1 nM T06273 C9T8PG 11680856 IC50 = 27 nM T06273 CCWE91 11726399 Ki = 0.376 nM T06273 C5F2AD 11760507 IC50 = 150 nM T06273 CE5HP1 11773441 EC50 = 400 nM T06273 CNLS20 11781868 IC50 = 173 nM T06273 CQB1H9 11807998 Ki = 7 nM T06273 CACX26 11808931 Ki = 263 nM T06273 CQ5PU0 11812259 IC50 = 134 nM T06273 CD8I3L 11817080 Ki = 692 nM T06273 CVKJ76 11822754 Ki = 9 nM T06273 C2PG3B 11832254 Ki = 7 nM T06273 CV8C4B 11832752 Ki = 57 nM T06273 CECF45 11833682 Ki = 10 nM T06273 CGU16R 11842604 EC50 = 3 nM T06273 CB3XT7 11842605 Ki = 19 nM T06273 CC7W8B 11959733 Ki = 23 nM T06273 CN50RE 11959814 EC50 = 3 nM T06273 C5D7HR 11959816 EC50 = 9 nM T06273 CE4UD7 11959906 EC50 = 2 nM T06273 CS0Z8U 11959909 EC50 = 4 nM T06273 CO6K5B 11959911 Ki = 870 nM T06273 CHFR46 11959914 Ki = 25 nM T06273 CMCB39 11960017 Ki = 25 nM T06273 C8X0GD 11960105 Ki = 32 nM T06273 CFW2E9 11960106 Ki = 45 nM T06273 C5YGB3 11960108 Ki = 50 nM T06273 C5SYR7 11960109 Ki = 41 nM T06273 CG9A1O 11960189 Ki = 24 nM T06273 C3Q6OZ 11960191 Ki = 12 nM T06273 C1EH9D 11960192 Ki = 33 nM T06273 C30KEW 11960193 Ki = 53 nM T06273 CGH8N3 11960194 Ki = 35 nM T06273 CEKX21 11960287 Ki = 140 nM T06273 C5S6TX 11960528 EC50 = 3 nM T06273 CI0QP9 11960529 IC50 = 1 nM T06273 CP0W7H 11960530 EC50 = 3 nM T06273 C97TSZ 11960533 EC50 = 4 nM T06273 C36ESI 11960630 EC50 = 6 nM T06273 CY1D6C 11960631 Ki = 4 nM T06273 C8UWV1 11960635 EC50 = 2 nM T06273 C3JD5M 11960733 EC50 = 2 nM T06273 C8LDK9 11960735 Ki = 13 nM T06273 CR1Z8W 11960736 EC50 = 18 nM T06273 C61QWS 11960831 Ki = 4 nM T06273 CP0HL6 11960919 EC50 = 2 nM T06273 C3RSB6 11960920 EC50 = 5 nM T06273 C7J8ME 11960923 EC50 = 8 nM T06273 C3VTN1 11960925 Ki = 3 nM T06273 C6IO2N 11960926 EC50 = 2 nM T06273 CA21PV 11961002 EC50 = 4 nM T06273 CUR0P8 11961006 EC50 > 1000 nM T06273 C7JK8Y 11961010 EC50 = 4 nM T06273 CIL6Z8 11961092 EC50 = 2 nM T06273 C7Y8MZ 12342815 IC50 = 311 nM T06273 CO03UJ 12407724 IC50 = 890 nM T06273 CH3I5Y 12494569 IC50 > 60000 nM T06273 CKDI53 12988985 IC50 = 30 nM T06273 CQM30I 13521672 IC50 > 100000 nM T06273 C1Y5AK 13815303 IC50 = 850 nM T06273 C06MRV 15488572 IC50 = 128 nM T06273 C2U4TR 15507355 IC50 = 100000 nM T06273 CG5A7W 16013152 IC50 > 19000 nM T06273 CBMF65 16013184 IC50 > 19000 nM T06273 C6V4TG 16013186 IC50 > 19000 nM T06273 CJ2XS5 16031314 IC50 = 55300 nM T06273 CFKO49 16216718 IC50 = 25 nM T06273 CSB5T2 16356047 IC50 = 1100 nM T06273 CGB34L 16357171 IC50 = 600 nM T06273 C9OC8G 16545097 IC50 = 820 nM T06273 CK6BD7 16665391 Ki = 2 nM T06273 COW9F1 16665466 Ki = 4 nM T06273 C5E2DM 16665467 EC50 = 2 nM T06273 CR8FW9 16665469 EC50 = 8 nM T06273 CAM95L 16665470 Ki = 3 nM T06273 C2E3GK 16665471 Ki = 12 nM T06273 C1I2OX 16665472 Ki = 4 nM T06273 CVP67B 16665552 EC50 = 6 nM T06273 CKN95X 16665623 Ki = 7 nM T06273 C8XSI5 16665626 EC50 = 7 nM T06273 C0JWR8 16665698 EC50 = 6 nM T06273 CV0W5R 16665702 Ki = 3 nM T06273 CN01VZ 16665773 Ki = 6 nM T06273 CB85MS 16665775 EC50 = 4 nM T06273 C79ROY 16665776 EC50 = 4 nM T06273 C4E1DM 16665847 Ki = 9 nM T06273 CR0H9Q 16665848 Ki = 2 nM T06273 CYQ1W3 16665853 Ki = 3 nM T06273 C70ZQK 16665934 EC50 = 1 nM T06273 CCA86L 16666013 Ki = 2 nM T06273 CMF5T4 16666250 EC50 = 1 nM T06273 C4CA2L 16666332 Ki = 4 nM T06273 CUS7D1 16666333 Ki = 1 nM T06273 C94YGN 17408065 IC50 = 280 nM T06273 CP32BE 17465122 IC50 = 1860 nM T06273 C0JQP8 17488605 IC50 = 49.8 nM T06273 CZWI52 17517933 IC50 = 1520 nM T06273 C4CXZ2 17564466 IC50 = 760 nM T06273 CR1PZ5 17567838 IC50 = 130 nM T06273 C5QJT3 17792611 IC50 = 100000 nM T06273 CLQO58 18428022 Ki = 26 nM T06273 C3JSU5 18428039 EC50 = 3 nM T06273 CN4Y8E 18428049 EC50 = 4 nM T06273 CF8J0L 18428130 EC50 = 4 nM T06273 CQ20JZ 18428167 Ki = 4 nM T06273 CA8HR9 18428182 EC50 = 12 nM T06273 CIE8Y3 18428218 EC50 = 9 nM T06273 CQ1SM3 18428266 Ki = 35 nM T06273 CDYJ74 18444338 IC50 = 9.5 nM T06273 C9UA1Y 18444343 IC50 = 13 nM T06273 CVR5M2 18444350 IC50 = 180 nM T06273 C95YGP 18444370 IC50 = 120 nM T06273 C2D1AI 18672397 IC50 = 100000 nM T06273 CGE9Z6 18676135 Ki = 7.2 nM T06273 C5X4BQ 18676146 Ki = 10.2 nM T06273 CEHQ15 18676147 Ki = 5.9 nM T06273 CX21CK 18676162 Ki = 5.6 nM T06273 CID4W5 18921977 IC50 = 2500 nM T06273 CWMC57 18973266 IC50 > 100000 nM T06273 C6IG3J 18973402 IC50 = 5030 nM T06273 CC2U8W 18973540 IC50 = 3070 nM T06273 CC8D1F 18973566 IC50 > 100000 nM T06273 C47JEK 19963762 IC50 = 9450 nM T06273 CB9I0W 20254879 IC50 > 19000 nM T06273 C8AX9U 20779872 IC50 = 299 nM T06273 C2M0NH 20779947 IC50 = 97 nM T06273 CVQ0W4 20779958 IC50 = 161 nM T06273 C5P0SC 20854918 IC50 = 5300 nM T06273 CZ6M5I 22431503 IC50 > 5011.87 nM T06273 CP9H4Y 22432631 IC50 > 5011.87 nM T06273 CG4H0A 22918383 IC50 = 2220 nM T06273 C54GJM 23624268 IC50 = 1.8 nM T06273 CL5O9X 23642205 EC50 = 230 nM T06273 CL0DF6 23705998 EC50 = 625 nM T06273 C9BL7H 24663409 IC50 = 280 nM T06273 C1LF9N 24764972 IC50 = 40 nM T06273 C90EOH 24771898 EC50 = 4600 nM T06273 C32SZN 24771899 EC50 = 2800 nM T06273 C28DRW 24771902 EC50 = 1400 nM T06273 CXF9H6 24771905 EC50 = 280 nM T06273 C3HU8I 24771951 IC50 = 0.5 nM T06273 CEC6K7 24771954 IC50 = 6 nM T06273 CZ6C0U 24771955 EC50 = 1600 nM T06273 CLE4T0 24771956 IC50 = 6 nM T06273 CC43TF 24771957 IC50 = 15 nM T06273 CN38TM 24771959 EC50 = 3200 nM T06273 CX4WH5 24772008 EC50 = 660 nM T06273 CDW8J1 24772009 EC50 = 200 nM T06273 C4A0VL 24772010 IC50 = 16 nM T06273 C1Y2MX 24772013 IC50 = 6 nM T06273 CWX0Q8 24772065 EC50 = 440 nM T06273 CUM6L9 24772069 EC50 = 420 nM T06273 CTE96I 24772070 EC50 = 310 nM T06273 CP9V4B 24772196 IC50 = 130 nM T06273 CNPV38 24772197 IC50 = 50 nM T06273 CQ69AN 24772641 EC50 = 2700 nM T06273 C9DKR6 24772642 IC50 = 12 nM T06273 C2NLG7 24772643 EC50 = 5200 nM T06273 C6IJ0N 24772644 IC50 = 14 nM T06273 C9W6AJ 24772646 IC50 = 7 nM T06273 CXAW15 24772712 EC50 = 260 nM T06273 CLTO20 24772713 IC50 = 4 nM T06273 CFY74R 24772716 IC50 = 11 nM T06273 CD6I1W 24772777 EC50 = 650 nM T06273 C5Q2GV 24772778 EC50 = 1100 nM T06273 CVMG41 24772779 EC50 = 900 nM T06273 C1NFY3 24772828 EC50 = 1300 nM T06273 C1AHW9 24772831 IC50 = 4 nM T06273 CFT10E 24772832 EC50 = 3500 nM T06273 CL8Q0K 24772834 IC50 = 1 nM T06273 CYE64C 24821029 IC50 = 3.8 nM T06273 C4GJ5U 24821031 IC50 = 3.1 nM T06273 CQXM45 24822105 IC50 = 3.7 nM T06273 C8NZ1F 24822107 IC50 = 2.6 nM T06273 C0XAH9 24822109 IC50 = 4.5 nM T06273 CI7R6L 24849157 Ki = 5 nM T06273 CQMW58 24851771 IC50 = 60 nM T06273 CLY1B7 24851881 IC50 = 230 nM T06273 C7EO6T 24851883 IC50 = 44 nM T06273 C1A9VR 24851885 IC50 = 45 nM T06273 CT0BP4 24852003 IC50 = 100 nM T06273 CC5O8P 24852124 IC50 = 97 nM T06273 C96SVC 24852130 IC50 = 27 nM T06273 C5WQE0 24852132 IC50 = 25 nM T06273 CI7U8M 24937579 Ki = 261 nM T06273 C4SLU7 24937580 Ki = 112 nM T06273 CTD51K 24937581 Ki = 391 nM T06273 CX9ET3 24937582 Ki = 123 nM T06273 C5L7GK 24937584 Ki > 9500 nM T06273 CQ2Y0A 24937701 EC50 = 53 nM T06273 CV2E4K 24937702 Ki = 32 nM T06273 C6AQ4S 24937703 Ki = 384 nM T06273 CPCE49 24937704 Ki = 164 nM T06273 C2X8JN 24937705 Ki = 140 nM T06273 CQB41I 24937706 Ki = 70 nM T06273 CM2KU7 24937834 Ki = 59 nM T06273 CP9IL2 24937836 Ki = 33 nM T06273 CB17QM 24937837 EC50 = 374 nM T06273 CO6M5C 24958198 IC50 = 3.2 nM T06273 C95FSV 24958199 IC50 = 2.4 nM T06273 CO28HF 25002578 Ki = 118 nM T06273 CK07MV 25002579 Ki = 3 nM T06273 C42NFR 25002581 Ki = 6 nM T06273 CTC24D 25002583 Ki = 112 nM T06273 CQ42OF 25002931 Ki = 6 nM T06273 C1O3RK 25002933 Ki = 9 nM T06273 CJR74F 25002935 Ki = 1.4 nM T06273 C7UPB2 25003288 Ki = 12 nM T06273 CVBA42 25003289 Ki = 4 nM T06273 CZB31N 25003291 Ki = 1.3 nM T06273 CXVR05 25003293 Ki = 14 nM T06273 C0IOR9 25015515 IC50 = 144.54 nM T06273 C3OVY8 25067330 IC50 = 100000 nM T06273 C63DJG 25117637 Ki = 0.9 nM T06273 CU3F7Y 25117638 Ki = 1.2 nM T06273 C5Z8BW 25119423 Ki = 1.6 nM T06273 CS2QU9 25120129 Ki = 0.9 nM T06273 C2YIX5 25122250 Ki = 1.3 nM T06273 C6ZC5I 25122604 Ki = 0.7 nM T06273 C8XPM1 25122606 Ki = 1.2 nM T06273 C5C8AR 25122607 Ki = 0.4 nM T06273 CJF4W8 25122608 Ki = 1.2 nM T06273 C06NFW 25122972 Ki = 6 nM T06273 C8JM9A 25122977 Ki = 0.4 nM T06273 CEQ70R 25128834 IC50 = 2 nM T06273 C8JEB3 25132256 IC50 = 9 nM T06273 CI9D5L 25132257 IC50 = 18 nM T06273 C0SG5U 25132258 IC50 = 7 nM T06273 CZ2V6U 25132259 IC50 = 18 nM T06273 CQ7GN6 25132260 IC50 = 23 nM T06273 C3FKN1 25132261 IC50 = 20 nM T06273 CFMS12 25132609 IC50 = 8 nM T06273 C83RAS 25132610 IC50 = 12 nM T06273 COP94S 25132611 IC50 = 12 nM T06273 CF3UY8 25132612 IC50 = 30.5 nM T06273 C7UV1Z 25132613 IC50 = 10 nM T06273 C5ABS6 25132952 IC50 = 2 nM T06273 C50JYL 25132953 IC50 = 2 nM T06273 CFN61R 25132954 IC50 = 3 nM T06273 C4FJ1R 25132955 IC50 = 12 nM T06273 CPJK86 25132956 IC50 = 8 nM T06273 CQR74H 25132957 IC50 = 8 nM T06273 CEP75B 25133278 IC50 = 6 nM T06273 CS45AM 25133279 IC50 = 51 nM T06273 C89NTJ 25133280 IC50 = 5 nM T06273 CB74VH 25133281 IC50 = 11 nM T06273 C0ZA1E 25133282 IC50 = 6 nM T06273 CW1R6V 25133283 IC50 = 39 nM T06273 CR28JV 25133629 IC50 = 12 nM T06273 C0XSY1 25133630 IC50 = 88 nM T06273 CRD2P8 25133631 IC50 = 13 nM T06273 C34UGQ 25133632 IC50 = 6 nM T06273 C4K2YL 25133633 IC50 = 6 nM T06273 C8GUM0 25133634 IC50 = 5 nM T06273 CY5JM6 25133974 IC50 = 4 nM T06273 C36AON 25133975 IC50 = 6 nM T06273 C2FKV0 25133976 IC50 = 5 nM T06273 CS69UT 25133977 IC50 = 2 nM T06273 C3XB9A 25133978 IC50 = 3 nM T06273 C27UDC 25133979 IC50 = 15 nM T06273 C24KEB 25143886 IC50 = 140 nM T06273 CNFC98 25156001 Ki = 37 nM T06273 CS9P5T 25156002 Ki = 9 nM T06273 C6O9QE 25156005 EC50 = 14 nM T06273 C6YK3O 25156006 Ki = 161 nM T06273 CBF17T 25156280 EC50 = 25 nM T06273 CT3MY8 25156282 EC50 = 29 nM T06273 CBJF14 25156286 EC50 = 31 nM T06273 CX4Q0V 25156561 Ki = 280 nM T06273 C0L5YX 25190716 Ki = 34 nM T06273 CWIQ61 25190717 Ki = 6 nM T06273 C9U6QF 25190718 Ki = 7 nM T06273 C2B1KZ 25190719 EC50 = 16 nM T06273 COA4P3 25190720 EC50 = 29 nM T06273 C1JFN2 25190721 EC50 = 14 nM T06273 C2P7NK 25190722 Ki = 5 nM T06273 CB0H8V 25190723 Ki = 110 nM T06273 CSK6M5 25190724 Ki = 180 nM T06273 C4TYE2 25190725 EC50 = 16 nM T06273 CIT27Q 25190726 Ki = 15 nM T06273 CN4J5V 25190727 Ki = 8 nM T06273 CWU16N 25190728 Ki = 26 nM T06273 CUIO49 25190729 EC50 = 12 nM T06273 CBZ92Q 25190730 EC50 = 15 nM T06273 CEV5A3 25190731 EC50 = 2 nM T06273 C51UAK 25190732 EC50 = 6 nM T06273 CZL3N9 25190733 Ki = 29 nM T06273 CM1P7G 25190734 EC50 = 13 nM T06273 CP3Z2W 25190735 EC50 = 5 nM T06273 C5VUQ3 25190736 Ki = 3 nM T06273 CRFS16 25190737 Ki = 5 nM T06273 CQ2M0Y 25190738 EC50 = 1 nM T06273 C7UTZ4 25190739 Ki = 16 nM T06273 CS8KG2 25190740 Ki = 27 nM T06273 C5F4JK 25190741 Ki = 28 nM T06273 CP5U2F 25190742 Ki = 31 nM T06273 CIQ8S9 25190743 EC50 = 9 nM T06273 CDR5U2 25190744 EC50 = 21 nM T06273 CYX8L2 25190745 EC50 = 13 nM T06273 CE1AK4 25190746 EC50 = 25 nM T06273 C09IBH 25190747 EC50 = 67 nM T06273 CXJ51W 25190748 EC50 = 3 nM T06273 C8T5DJ 25190749 EC50 = 1 nM T06273 C02EPW 25190750 EC50 = 7 nM T06273 C7H3CA 25190751 EC50 = 20 nM T06273 CPIK86 25190752 Ki = 4 nM T06273 CV72DI 25190930 IC50 = 300 nM T06273 CR01KW 25208411 IC50 = 240 nM T06273 CT1JU9 25208412 IC50 = 4533 nM T06273 C04LVZ 25208413 IC50 = 12399 nM T06273 CJSV48 25208414 IC50 = 9332 nM T06273 CH63ZF 25208597 IC50 = 52000 nM T06273 C93LPA 25208906 IC50 = 62000 nM T06273 C7CGB8 25208907 IC50 = 43000 nM T06273 CVK43I 25209053 IC50 = 27000 nM T06273 CNOV-37 25209059 IC50 = 23000 nM T06273 C0KQ3B 25218483 IC50 = 8 nM T06273 CT18QY 25218484 IC50 = 5 nM T06273 CE29IV 25218485 IC50 = 18 nM T06273 COZ07N 25218486 IC50 = 61 nM T06273 CT34JM 25218487 IC50 = 24 nM T06273 CBHS06 25218488 IC50 = 50 nM T06273 CUS9Q3 25218489 IC50 = 970 nM T06273 CP1N6Y 25218490 IC50 > 10000 nM T06273 CMSN20 25218491 IC50 = 200 nM T06273 COG2Q9 25218492 IC50 = 103 nM T06273 C0ACL6 25218493 IC50 = 200 nM T06273 C7D3AV 25218494 IC50 = 19 nM T06273 C94ORH 25218495 IC50 = 29 nM T06273 CE80FZ 25218496 IC50 = 240 nM T06273 CXCM83 25218497 IC50 = 250 nM T06273 CMK80A 25218498 IC50 = 1500 nM T06273 CQF12I 25218499 IC50 > 10000 nM T06273 C1CNI5 25218500 IC50 = 12 nM T06273 C15BZH 25218501 IC50 = 14 nM T06273 CCBA43 25589747 IC50 = 350 nM T06273 CQL5P7 26160509 IC50 = 3715.35 nM T06273 CUJ06V 26676715 IC50 = 87.6 nM T06273 C0ADR6 26828969 IC50 = 1060 nM T06273 C9WB0S 27319973 IC50 = 820 nM T06273 CMXA39 28825277 IC50 > 100000 nM T06273 CSO1Z6 28825295 IC50 > 100000 nM T06273 CF7RU3 37346305 IC50 = 2540 nM T06273 CG98XO 40152038 IC50 < 13000 nM T06273 C9H4YK 42605457 IC50 = 45 nM T06273 CM4S1W 42605563 IC50 = 99 nM T06273 CNH4I3 42605667 IC50 = 536 nM T06273 C73CSQ 42605668 IC50 = 78 nM T06273 CGN73X 42605896 IC50 = 8 nM T06273 C7UY8H 42606009 IC50 = 60 nM T06273 C6UYV0 42606011 IC50 = 36 nM T06273 C4O1WX 42606017 IC50 = 234 nM T06273 CG7U8W 42606131 IC50 = 175 nM T06273 C6EF0Z 42606133 IC50 = 188 nM T06273 CTR6N9 42606240 IC50 = 187 nM T06273 CIZY42 42606242 IC50 = 47 nM T06273 CW69VT 42606249 IC50 = 40 nM T06273 C8W7QG 42606356 IC50 = 19 nM T06273 C08QIG 42606362 IC50 = 44 nM T06273 C96QNS 42606476 IC50 = 30 nM T06273 CZ07WD 42606478 IC50 = 65 nM T06273 CW3TC5 42606480 IC50 = 42 nM T06273 C6IFE0 42606484 IC50 = 79 nM T06273 CWVU62 42606592 IC50 = 134 nM T06273 CG47NA 42606596 IC50 = 166 nM T06273 CUMV68 42606602 IC50 = 68 nM T06273 CF1X4W 42606708 IC50 = 67 nM T06273 CQFB09 42606718 IC50 = 71 nM T06273 CI6H2M 42606720 IC50 = 42 nM T06273 C52QRE 42606833 IC50 = 40 nM T06273 CXDQ78 42606835 IC50 = 173 nM T06273 C4ZP8N 42606948 IC50 = 28 nM T06273 C21ZSK 42606950 IC50 = 39 nM T06273 C40EUZ 42606952 IC50 = 80 nM T06273 C9PCL3 42606954 IC50 = 56 nM T06273 C0SOE4 42607057 IC50 = 25 nM T06273 C6PL3B 42607059 IC50 = 13 nM T06273 CETP17 42607061 IC50 = 53 nM T06273 C6N7ET 42607064 IC50 = 695 nM T06273 CH5KC6 42607170 IC50 = 38 nM T06273 CZ1IN0 42888548 IC50 = 1960 nM T06273 CBH1S5 44251671 IC50 = 35 nM T06273 CC3VN4 44291540 IC50 = 57 nM T06273 C3OIC9 44291541 IC50 = 184 nM T06273 CX5R6W 44291587 IC50 > 100000 nM T06273 CKT58E 44291868 IC50 = 14000 nM T06273 CI85LY 44291869 IC50 = 36 nM T06273 CGV0U4 44292001 IC50 = 195 nM T06273 CTE7Q6 44292099 IC50 = 21 nM T06273 CRZ93Q 44292100 IC50 = 136 nM T06273 CQB02S 44292118 IC50 = 92 nM T06273 C2K5VF 44317843 Ki = 4.5 nM T06273 C15CVA 44317906 Ki = 12 nM T06273 C0VA2H 44318172 IC50 = 42 nM T06273 C1CEF0 44318206 IC50 = 31 nM T06273 CNF2V0 44318316 IC50 = 243 nM T06273 CS23CF 44318317 IC50 = 116 nM T06273 CS5K8T 44318336 IC50 = 210 nM T06273 C16DOS 44318591 IC50 = 349 nM T06273 CG5D9Z 44318603 IC50 = 185 nM T06273 CAG93U 44318616 IC50 = 99 nM T06273 CE3XT5 44318617 IC50 = 240 nM T06273 CTS7Z1 44336824 IC50 = 51 nM T06273 CZC24Y 44336846 IC50 = 112 nM T06273 C0WGR7 44337636 EC50 = 400 nM T06273 C4VZK2 44337637 IC50 = 12 nM T06273 CA23WF 44337647 IC50 = 15 nM T06273 CS8M6G 44337900 IC50 = 450 nM T06273 CB9L3C 44337901 EC50 = 200 nM T06273 CVY63H 44337902 IC50 = 15 nM T06273 C8S5CE 44337906 IC50 = 12 nM T06273 CHEN95 44337964 IC50 > 5000 nM T06273 CZKB70 44337977 IC50 = 50 nM T06273 CSM7C1 44337979 EC50 = 80 nM T06273 CDI7H4 44337980 IC50 = 400 nM T06273 CSQ12W 44337988 IC50 = 20 nM T06273 C5ZY1U 44337990 EC50 = 2000 nM T06273 CF6LY9 44338005 IC50 = 900 nM T06273 CFZ39L 44338020 IC50 = 150 nM T06273 C35EPF 44338034 IC50 = 3000 nM T06273 CPT3C1 44338036 IC50 = 250 nM T06273 CRN78F 44338056 IC50 = 60 nM T06273 CBTZ12 44338066 EC50 = 300 nM T06273 CD3MF7 44338072 EC50 = 700 nM T06273 CWSD01 44338073 IC50 = 40 nM T06273 C8AM7O 44338076 IC50 > 5000 nM T06273 C0Z3PL 44338078 IC50 = 900 nM T06273 C0A5ZQ 44338090 IC50 = 40 nM T06273 CK91NC 44338091 IC50 = 800 nM T06273 CCL2R8 44338129 IC50 = 200 nM T06273 CLU41A 44338185 IC50 = 70 nM T06273 CS2C8D 44338198 EC50 = 100 nM T06273 CRAP20 44338202 EC50 = 900 nM T06273 C64OEZ 44338216 IC50 = 60 nM T06273 CAT5W0 44338228 EC50 = 200 nM T06273 C2NE1F 44338230 IC50 = 30 nM T06273 CCHV95 44338243 IC50 = 30 nM T06273 C5P6XV 44338244 IC50 = 20 nM T06273 CJ2U6W 44338275 IC50 = 300 nM T06273 C83AJW 44338282 IC50 = 3000 nM T06273 CMY2O1 44338295 IC50 = 25 nM T06273 CM75XU 44338296 IC50 = 30 nM T06273 CGI73S 44338474 EC50 = 70 nM T06273 C61EFU 44363892 Ki = 6 nM T06273 CX40WQ 44363946 Ki = 10 nM T06273 C56UTP 44363947 Ki = 23 nM T06273 C8BKV6 44381234 IC50 = 45 nM T06273 CW2D0G 44396612 Ki = 6.8 nM T06273 CCG08R 44396740 Ki = 12.5 nM T06273 CF7T8X 44396942 Ki = 87 nM T06273 C1DLG3 44401996 IC50 = 36 nM T06273 CA17OQ 44401997 IC50 = 90 nM T06273 CU0V4C 44402080 IC50 = 13 nM T06273 CC51DW 44402081 IC50 = 116 nM T06273 CV18CA 44402096 IC50 = 90 nM T06273 C8I9OL 44402097 IC50 = 370 nM T06273 C6D0UG 44402115 IC50 = 47 nM T06273 CE5JY1 44402125 IC50 = 9.8 nM T06273 C37DOY 44402155 IC50 = 50 nM T06273 CF1AN8 44402172 IC50 = 56 nM T06273 CU89YV 44402216 IC50 = 10 nM T06273 CNR89L 44402230 IC50 = 20 nM T06273 C07JOB 44402244 IC50 = 290 nM T06273 CA42ZV 44402245 IC50 = 189 nM T06273 C36TFA 44402292 IC50 = 55 nM T06273 CP02AG 44402324 IC50 = 27 nM T06273 CG08PV 44402327 IC50 = 540 nM T06273 C23YOE 44403364 IC50 = 249 nM T06273 CLIN21 44403373 IC50 = 495 nM T06273 CPNS90 44403374 IC50 = 8.9 nM T06273 CY3VP2 44403382 IC50 = 8600 nM T06273 CAN85F 44403383 IC50 = 200 nM T06273 COW1U4 44403389 IC50 = 6100 nM T06273 C6WLC7 44403390 IC50 = 274 nM T06273 C2QT9O 44403395 IC50 > 10000 nM T06273 C0M8YG 44403396 IC50 = 467 nM T06273 CGD03T 44407483 IC50 = 15 nM T06273 CM21WK 44407525 IC50 = 10000 nM T06273 C3RP9B 44407531 IC50 = 6 nM T06273 CFW6D5 44407532 IC50 = 16 nM T06273 CGC50I 44407533 IC50 > 10000 nM T06273 CB8VK7 44407534 IC50 > 10000 nM T06273 CU53QL 44407535 IC50 > 10000 nM T06273 C0RF8K 44407537 IC50 = 8 nM T06273 CQB73J 44407559 IC50 = 15 nM T06273 C6GL3U 44407567 IC50 > 10000 nM T06273 CZVS93 44407569 IC50 = 9 nM T06273 CCK6X0 44407570 IC50 = 16 nM T06273 CU0H6W 44407571 IC50 = 56 nM T06273 C7GV4H 44407572 IC50 = 8 nM T06273 C2S6GO 44407702 IC50 = 46 nM T06273 C5R6UB 44407737 IC50 = 40 nM T06273 C0MB3L 44407780 IC50 = 15 nM T06273 C16SHL 44407781 IC50 = 8 nM T06273 CR7C8H 44407793 IC50 = 9 nM T06273 C5E0JM 44407794 IC50 = 8 nM T06273 C2IBO3 44407795 IC50 = 10000 nM T06273 C02JPH 44407888 IC50 = 9 nM T06273 CM18QR 44407895 IC50 = 7 nM T06273 C4E6BF 44407931 IC50 = 5 nM T06273 CYIJ34 44407937 IC50 = 10 nM T06273 CZ2N6P 44407942 IC50 = 6 nM T06273 CUVG05 44407993 IC50 = 14 nM T06273 C9PKN0 44408006 IC50 = 5 nM T06273 CG8KJ4 44408056 IC50 = 8 nM T06273 C8H3CF 44408057 IC50 = 23 nM T06273 C1VHS7 44408064 IC50 = 15 nM T06273 C8BR0A 44408065 IC50 = 5 nM T06273 CCP9G2 44408105 IC50 = 12 nM T06273 CWEQ40 44408111 IC50 = 8 nM T06273 CW3JX5 44408115 IC50 = 9 nM T06273 C2KL9I 44408130 IC50 = 10000 nM T06273 CM7U9T 44408131 IC50 = 3000 nM T06273 CM2IG6 44408192 IC50 = 162 nM T06273 C47ERA 44408194 IC50 = 83 nM T06273 CAS7G8 44408200 IC50 = 65 nM T06273 CV9OH6 44408203 IC50 = 237 nM T06273 CK5WS6 44408204 IC50 = 161 nM T06273 CC4AO9 44408236 IC50 = 30 nM T06273 CZQS73 44408237 IC50 = 18 nM T06273 CBC29E 44408241 IC50 = 200 nM T06273 C7DK0R 44408242 IC50 = 80 nM T06273 C1X5VO 44408243 IC50 = 59 nM T06273 C10OYN 44408244 IC50 = 120 nM T06273 C0JBR4 44408250 IC50 = 165 nM T06273 CVN7C1 44408277 IC50 = 105 nM T06273 C7NX5U 44408348 IC50 = 670 nM T06273 CDG10Z 44408373 IC50 = 80 nM T06273 CC1BG3 44440323 IC50 = 40 nM T06273 C0V5SN 44440326 IC50 = 84 nM T06273 CBT7H1 44440329 IC50 = 42 nM T06273 CQ54RI 44440331 IC50 = 20 nM T06273 C81ZTJ 44440332 IC50 = 56 nM T06273 C4U0RW 44440339 IC50 = 42 nM T06273 C8Z7MP 44440340 IC50 = 32 nM T06273 CUM65V 44440341 IC50 = 56 nM T06273 C5Y1IZ 44440342 IC50 = 56 nM T06273 CRA7C0 44440344 IC50 = 49 nM T06273 CQV98J 44440345 IC50 = 52 nM T06273 CI15DF 44440347 IC50 = 20 nM T06273 CJD3Q8 44440349 IC50 = 18 nM T06273 CLGH28 44440351 IC50 = 20 nM T06273 CNA3D4 44440352 IC50 = 50 nM T06273 C72NQF 44440353 IC50 = 54 nM T06273 CCP5K1 44440354 IC50 = 19 nM T06273 C9IE6K 44440355 IC50 = 54 nM T06273 CH7K2Q 44440356 IC50 = 46 nM T06273 CJ95HX 44440361 IC50 = 22 nM T06273 CLC87O 44440364 IC50 = 38 nM T06273 C4U9MB 44440366 IC50 = 21 nM T06273 CEH05M 44440371 IC50 = 29 nM T06273 C79KRC 44440377 IC50 = 60 nM T06273 C2Z7NT 44440379 IC50 = 66 nM T06273 CR8GT3 44440380 IC50 = 17 nM T06273 CE7Y5R 44460202 Ki = 8.7 nM T06273 CI5EV2 44460224 Ki = 5.9 nM T06273 CK6IW9 44460253 Ki = 31 nM T06273 CR4D8E 44460362 Ki = 9.8 nM T06273 C3FJA7 44460520 Ki = 11.7 nM T06273 CNL10E 44460532 Ki = 272 nM T06273 CW43EB 44473424 Ki = 1 nM T06273 CNI3Y5 44483163 IC50 > 18700 nM T06273 C2PJM6 44541767 Ki = 1.2 nM T06273 CFZA14 44541770 Ki = 2.4 nM T06273 C4G2XV 44541771 Ki = 6.8 nM T06273 C6PHU3 44541772 Ki = 4 nM T06273 CG69PI 44541773 Ki = 20 nM T06273 CUX7G1 44541918 Ki = 10 nM T06273 C10RXH 44541919 Ki = 4.5 nM T06273 C1TPI7 44541920 Ki = 0.95 nM T06273 C1ZCT3 44541922 Ki = 0.76 nM T06273 CJ5P6Q 44541924 EC50 = 2.2 nM T06273 CB8QP4 44542060 Ki = 2.9 nM T06273 CV93DX 44542063 Ki = 1.6 nM T06273 C8NH1A 44542066 Ki = 2 nM T06273 CZD12F 44542210 Ki = 1.7 nM T06273 CJ82YH 44542211 Ki = 2.2 nM T06273 C5OUF2 44542363 Ki = 3.8 nM T06273 C3SOX5 44542366 Ki = 1.9 nM T06273 C5D6WY 44549376 IC50 = 2.2 nM T06273 CH0B8D 44549377 IC50 = 1.4 nM T06273 CSF25A 44549378 IC50 = 3.1 nM T06273 C6XO1Q 44549379 IC50 = 9 nM T06273 C06EWM 44549510 IC50 = 270 nM T06273 CDB3E5 44549647 IC50 = 3.7 nM T06273 C8ZL1T 44549648 IC50 = 4.8 nM T06273 CXC7G4 44549649 IC50 = 1.9 nM T06273 CN3MI4 44549650 IC50 = 17 nM T06273 C48VTG 44549651 IC50 = 31 nM T06273 CV98BR 44549774 IC50 = 5.9 nM T06273 CSG41C 44549775 IC50 = 3.8 nM T06273 C2U7CB 44549776 IC50 = 4.3 nM T06273 C7HWK5 44549777 IC50 = 2.1 nM T06273 CIXL54 44549778 IC50 = 14 nM T06273 CT97YW 44549779 IC50 = 6.7 nM T06273 C3F9SI 44549780 IC50 = 3.7 nM T06273 C2ZD1T 44549902 IC50 = 16 nM T06273 CD0GB9 44549904 IC50 = 200 nM T06273 C2LC0O 44549906 IC50 = 5.3 nM T06273 C6JR0G 44567831 Ki = 61 nM T06273 C9B8ZY 44567867 Ki = 50 nM T06273 CFNJ45 44567901 Ki = 18 nM T06273 CP10ME 44567902 Ki = 58 nM T06273 C2SY5G 44567903 EC50 = 2 nM T06273 CF02VL 44567953 EC50 = 1.3 nM T06273 CDH8J6 44567954 EC50 = 1.8 nM T06273 C8CGB7 44567955 Ki = 19 nM T06273 C0L5GZ 44567956 Ki = 17 nM T06273 C52YBK 44567957 EC50 = 0.9 nM T06273 CE59GP 44568000 EC50 = 3.1 nM T06273 C7H5VI 44571000 IC50 = 25 nM T06273 CTY51E 44571001 IC50 = 46 nM T06273 C0ZC8K 44571087 IC50 = 45 nM T06273 C6RS8T 44571088 IC50 = 100 nM T06273 C2PT7V 44571133 IC50 = 27 nM T06273 C1Z5SH 44571256 IC50 = 109 nM T06273 CWSU12 44603416 IC50 = 470 nM T06273 C7DTS2 45084012 IC50 = 1000 nM T06273 CE3DV0 45267516 IC50 = 41 nM T06273 CMC10I 45268371 IC50 = 130 nM T06273 C7CB8Y 45268372 IC50 = 53 nM T06273 CA4WY0 45268384 IC50 = 120 nM T06273 CIA92V 45268393 IC50 = 58 nM T06273 CH8PY5 45268394 IC50 = 390 nM T06273 C8OF3J 45268634 Ki = 239 nM T06273 CBA0Z7 45268640 Ki = 190 nM T06273 C40DSP 45269234 IC50 > 500 nM T06273 CQU91E 45269470 Ki = 23 nM T06273 CRY07G 45270081 IC50 = 82 nM T06273 C2JBZ4 45270088 IC50 = 110 nM T06273 CH85VZ 45270094 IC50 = 130 nM T06273 CC07DP 45270307 Ki = 149 nM T06273 CY2E0P 45270924 IC50 = 180 nM T06273 C5OL7C 45271137 Ki = 519 nM T06273 CX0I1K 45271138 Ki = 1120 nM T06273 CJC26X 45271143 EC50 = 39 nM T06273 C38SXR 45271764 IC50 = 340 nM T06273 CYI8P4 45272031 Ki = 589 nM T06273 CZP38X 45272044 Ki = 96 nM T06273 CO9AK7 45272045 EC50 = 58 nM T06273 C4HZN0 45272632 IC50 = 85 nM T06273 CZF4L5 45272633 IC50 > 500 nM T06273 C0VB6T 45272650 IC50 = 230 nM T06273 CN48FT 45272850 Ki = 133 nM T06273 C1DP9C 45273550 IC50 = 160 nM T06273 CU4HQ8 45273796 Ki = 698 nM T06273 C8V9PH 45273804 Ki = 23 nM T06273 CAM34R 45484114 Ki = 2 nM T06273 CBW72V 46173035 Ki = 6 nM T06273 C51MOF 46191765 IC50 = 4 nM T06273 C2YZK5 46205122 Ki = 3 nM T06273 C78HMZ 46206097 EC50 = 3 nM T06273 C2YL5D 46216737 IC50 = 1.3 nM T06273 CM82CZ 46216738 IC50 = 2.8 nM T06273 C8BN4H 46216788 IC50 = 2 nM T06273 C1AI8S 46216791 EC50 = 22 nM T06273 C57OFD 46216800 IC50 = 2.5 nM T06273 C7WNR9 46216801 IC50 = 3.6 nM T06273 C3JUH5 46216812 IC50 = 5.4 nM T06273 CQ4X2Z 46225750 IC50 > 100000 nM T06273 CM8CX2 46225751 IC50 = 14850 nM T06273 CL2I1K 46225752 IC50 = 12090 nM T06273 CV42SR 46225765 IC50 = 36 nM T06273 C42GQJ 46225772 IC50 = 5870 nM T06273 C1YFR9 46225777 IC50 > 100000 nM T06273 CHVG15 46225795 IC50 = 3230 nM T06273 CX2O4K 46225796 IC50 = 5780 nM T06273 C20ECV 46225797 IC50 = 4110 nM T06273 CZ80EI 46225801 IC50 = 3310 nM T06273 C3N1HC 46225802 IC50 = 4270 nM T06273 CIBA87 46225807 IC50 = 560 nM T06273 CV1A5K 46225808 IC50 > 100000 nM T06273 C81PFD 46226062 IC50 = 12 nM T06273 CB2DX8 46226063 IC50 = 6 nM T06273 CIFD31 46226065 IC50 = 13 nM T06273 CH6U5W 46226100 IC50 = 11 nM T06273 CV5K7N 46226101 IC50 = 4 nM T06273 CKW20Q 46226102 EC50 = 2800 nM T06273 CKI8G7 46226264 IC50 = 10 nM T06273 C23SHF 46226265 IC50 = 20 nM T06273 CP9E3K 46226266 IC50 = 38 nM T06273 CLNR34 46226282 IC50 = 54 nM T06273 CH5M9A 46226283 IC50 = 10 nM T06273 CB8Z6M 46226284 IC50 = 30 nM T06273 C2NK1X 46226285 IC50 = 22 nM T06273 C65LBF 46226286 IC50 = 40 nM T06273 C6BDU7 46226300 IC50 = 15 nM T06273 CKJ1S4 46226301 IC50 = 10 nM T06273 CJ7VP9 46226302 IC50 = 20 nM T06273 CB8IF9 46226303 IC50 = 30 nM T06273 CO7LS9 46226304 IC50 = 46 nM T06273 C6OHS2 46226326 IC50 = 10 nM T06273 CQ4VB7 46226327 IC50 = 30 nM T06273 CE9X6Y 46226328 IC50 = 20 nM T06273 C9JYF4 46226329 IC50 = 17 nM T06273 CVD2F9 46226330 IC50 = 10 nM T06273 CG5DH9 46226350 IC50 = 25 nM T06273 CPHZ76 46226351 IC50 = 18 nM T06273 C91AUJ 46226352 IC50 = 22 nM T06273 C3I2NP 46226353 IC50 = 65 nM T06273 CPQ5K0 46226354 IC50 = 5 nM T06273 C0P8FS 46226375 IC50 = 4 nM T06273 CE4W3M 46226376 IC50 = 12 nM T06273 CNES04 46226377 IC50 = 4 nM T06273 CUQ98E 46226378 IC50 = 20 nM T06273 CF0SI7 46226379 IC50 = 180 nM T06273 CNYR50 46226380 IC50 = 5 nM T06273 CF0W9T 46226381 IC50 = 37 nM T06273 C5HMG4 46226395 IC50 = 8 nM T06273 CGP48Z 46226396 IC50 = 1.4 nM T06273 CV6G4T 46226397 IC50 = 20 nM T06273 CMU91T 46226398 IC50 = 25 nM T06273 CHB6I9 46226399 IC50 > 1000 nM T06273 CKO2E1 46226401 IC50 = 35 nM T06273 CZT04Y 46226418 IC50 = 6 nM T06273 CLA2F9 46226419 IC50 = 2 nM T06273 CTJ04X 46226420 IC50 = 16 nM T06273 CJQ53X 46226421 IC50 = 5 nM T06273 CJXS95 46226422 IC50 = 6 nM T06273 C81DRT 46226423 EC50 = 1200 nM T06273 CZO4D2 46226424 EC50 = 1700 nM T06273 CZ0O5B 46229747 IC50 = 12 nM T06273 C40RUD 46229748 IC50 = 3.8 nM T06273 CU2T9B 46229749 IC50 = 1.8 nM T06273 C97APF 46229754 IC50 = 2.3 nM T06273 C61NYF 46229755 IC50 = 41 nM T06273 C54VHJ 46229756 IC50 = 6.3 nM T06273 C2SAO5 46229757 IC50 = 200 nM T06273 CJNP40 46229796 IC50 = 3.3 nM T06273 C74RCE 46229797 IC50 = 4.2 nM T06273 CSI85P 46229802 IC50 = 13 nM T06273 CFS86M 46229803 IC50 = 18 nM T06273 C9QJ3E 46229804 IC50 = 7.2 nM T06273 CP5MZ2 46229844 IC50 = 2.5 nM T06273 CL0EA1 46229848 IC50 = 24 nM T06273 CM21HU 46229849 IC50 = 2.8 nM T06273 CPW65M 46229850 IC50 = 3.1 nM T06273 C93BTO 46229851 IC50 = 0.7 nM T06273 CQJR19 46229887 IC50 = 14 nM T06273 CMG6Q1 46229888 IC50 = 15 nM T06273 C5H7YU 46229889 IC50 = 1.8 nM T06273 C20LYS 46229944 IC50 = 1 nM T06273 C4LF2J 46229945 IC50 = 7.1 nM T06273 CRSM18 46229946 IC50 = 2.6 nM T06273 C7ATR8 46229947 IC50 = 22 nM T06273 CR9A3Y 46229995 IC50 = 1 nM T06273 CCM7I4 46229996 IC50 = 6.2 nM T06273 C9P1JF 46230050 IC50 = 8.2 nM T06273 CGW5A0 46230051 IC50 = 9 nM T06273 C42MPI 46230223 IC50 = 9.7 nM T06273 CYT2P5 46230224 IC50 = 4.7 nM T06273 CR56WD 46230228 IC50 = 1 nM T06273 CV4S3F 46230229 IC50 = 2.6 nM T06273 CVY9X0 46230230 IC50 = 4 nM T06273 CZ47OW 46230231 IC50 = 59 nM T06273 CQ21YC 46230232 IC50 = 14 nM T06273 CP43OL 46230279 IC50 = 4.6 nM T06273 CGY96Q 46230280 IC50 = 1.8 nM T06273 CB90YW 46230281 IC50 = 3.6 nM T06273 COS16C 46230285 IC50 = 14 nM T06273 CF68UE 46230286 IC50 = 13 nM T06273 C1QPD5 46230287 IC50 = 3.2 nM T06273 C8OM4X 46230288 IC50 = 2.1 nM T06273 CBP81Q 46230327 IC50 = 5.7 nM T06273 CN49ZV 46230328 IC50 = 2.7 nM T06273 CL0ZQ2 46230329 IC50 = 3.1 nM T06273 CML89C 46230330 IC50 = 2.4 nM T06273 CL8ZR3 46230332 IC50 = 1 nM T06273 CC8ZD5 46230333 IC50 = 3.7 nM T06273 CAI80X 46230334 IC50 = 2.4 nM T06273 CQNS64 46230335 IC50 = 3.1 nM T06273 C2OE8J 46230372 IC50 = 2.7 nM T06273 CFRL41 46230373 IC50 = 3.9 nM T06273 CEL70I 46230374 IC50 = 3.5 nM T06273 CO8J7R 46230376 IC50 = 9 nM T06273 CFJ0G9 46230377 IC50 = 2.4 nM T06273 C6H5IJ 46230378 IC50 = 2 nM T06273 CTWR26 46230379 IC50 = 2.5 nM T06273 CJM95V 46230422 IC50 = 3.2 nM T06273 C1M9UT 46230426 IC50 = 5.1 nM T06273 CR5IM1 46230427 IC50 = 12 nM T06273 C4J9KH 46230428 IC50 = 1.4 nM T06273 C6VMR5 46230429 IC50 = 2.3 nM T06273 CW39NM 46230507 IC50 = 3.1 nM T06273 C0NKH5 46230508 IC50 = 2.7 nM T06273 CB6I3Y 46230509 IC50 = 2.8 nM T06273 C6X4PF 46230510 IC50 = 3.9 nM T06273 C7WI3A 46230515 IC50 = 1.6 nM T06273 CB1IG2 46230516 IC50 = 1.6 nM T06273 CW8XS7 46230517 IC50 = 5 nM T06273 CJH0A8 46230518 IC50 = 19 nM T06273 CW0UB7 46230562 Ki = 314 nM T06273 C68HVY 46884129 IC50 = 29 nM T06273 C1C7YG 46884210 IC50 > 10000 nM T06273 C4IY0M 46905385 IC50 = 42 nM T06273 C68MEF 46918658 IC50 = 983.4 nM T06273 CS0WI8 46918661 IC50 = 1371.4 nM T06273 CHEG10 46918686 IC50 = 1075.6 nM T06273 CH8B3S 46926923 IC50 = 33 nM T06273 C42TEY 49797033 IC50 = 800 nM T06273 C03SIZ 49798923 IC50 = 9.204 nM T06273 CECB91 49843530 IC50 = 27 nM T06273 CF91RS 49843531 IC50 = 40 nM T06273 CIU38A 49871952 IC50 = 640 nM T06273 CFT6V9 49873225 IC50 = 50 nM T06273 CU93DH 49873226 IC50 = 162 nM T06273 C7J0FP 49890275 IC50 = 1340 nM T06273 CWG2D4 49890340 IC50 = 7810 nM T06273 CUI4C3 49891173 IC50 = 4810 nM T06273 CEQG01 49891329 IC50 = 13950 nM T06273 CRE5B9 50941753 IC50 = 700 nM T06273 C9Q1IE 50941754 IC50 = 400 nM T06273 C1CT3V 50941755 IC50 = 60 nM T06273 C8B2VI 50942807 IC50 = 1900 nM T06273 CK19LI 50943015 IC50 = 150 nM T06273 CI3M6X 50943089 IC50 > 10000 nM T06273 C7DV9L 50943090 IC50 = 1600 nM T06273 C4G1LY 50943161 IC50 = 1100 nM T06273 C3CPR5 50943163 IC50 = 6000 nM T06273 C1V9KR 50943164 IC50 = 3000 nM T06273 CCY08V 50943240 IC50 = 9900 nM T06273 CAW1F9 50943244 IC50 = 100 nM T06273 CWP2H1 50943321 IC50 = 110 nM T06273 C4SB5E 50943479 IC50 = 40 nM T06273 C6NT4Y 52936671 IC50 = 230 nM T06273 C79MDT 52936672 IC50 = 16600 nM T06273 C1R0WZ 52936673 IC50 < 11000 nM T06273 CWY42J 52936674 IC50 = 8600 nM T06273 C6ZW2S 52936676 IC50 = 1600 nM T06273 C8G9IY 52936778 IC50 = 550 nM T06273 CVTK78 52936780 IC50 = 13900 nM T06273 C7RW3J 52936781 IC50 = 13400 nM T06273 CWQ81A 52936782 IC50 = 3000 nM T06273 CI20KJ 52936783 IC50 = 10700 nM T06273 CMJ81G 52936784 IC50 = 18000 nM T06273 COZ67W 52936785 IC50 = 11200 nM T06273 CNV71W 52936890 IC50 = 7600 nM T06273 CJDH42 52936891 IC50 = 31600 nM T06273 CNQL08 52936892 IC50 = 4500 nM T06273 CY0C6G 52936893 IC50 = 22400 nM T06273 CB18GT 52936894 IC50 > 80000 nM T06273 C7UB5J 52936895 IC50 > 100000 nM T06273 C6NH8P 52936896 IC50 > 50000 nM T06273 CKX0Z7 53387188 IC50 = 120000 nM T06273 CJ2YZ7 53391638 IC50 = 500000 nM T06273 CWF40I 56587957 IC50 > 100000 nM T06273 CP56DT 56641533 IC50 = 1279.7 nM T06273 C3NX9F 56641534 IC50 = 976.5 nM T06273 CK7C5L 56641536 IC50 = 138.5 nM T06273 CIX1W6 56650290 IC50 = 90 nM T06273 C1S3NU 56658116 IC50 = 78000 nM T06273 C3IGF0 56658117 IC50 = 66000 nM T06273 CV8B2N 56665040 IC50 = 123000 nM T06273 C2FB5M 56832570 IC50 = 1.7 nM T06273 CMI7H2 56832632 IC50 = 5000 nM T06273 C4MXT0 56833017 IC50 = 2 nM T06273 C1QB2J 56834916 IC50 = 12 nM T06273 CJ49IO 56834929 IC50 = 7 nM T06273 CW8L1A 57333526 IC50 = 6800 nM T06273 C4QHN0 57390502 IC50 = 19 nM T06273 CV39SI 57390503 IC50 = 12 nM T06273 CZL06B 57390504 IC50 = 16 nM T06273 CV27UL 57390505 IC50 = 26 nM T06273 C2EVT7 57390506 IC50 = 16 nM T06273 C5AZS3 57390508 IC50 = 22 nM T06273 CB97KP 57390509 IC50 = 13 nM T06273 C5X0IM 57392280 IC50 = 15 nM T06273 CEF54Q 57392281 IC50 = 13 nM T06273 C09IQW 57394038 IC50 = 2 nM T06273 C5VIH7 57395797 IC50 = 8 nM T06273 C72YWA 57397575 IC50 = 10 nM T06273 CYV59M 57397576 IC50 = 12 nM T06273 CIH09D 57399257 IC50 = 3 nM T06273 C3G4ZK 57401019 IC50 = 12 nM T06273 CURB16 57401020 IC50 = 10 nM T06273 CB2YO3 57401022 IC50 = 15 nM T06273 CQZ9U6 57401023 IC50 = 9 nM T06273 COKM60 57402780 IC50 = 7 nM T06273 CDE07O 60150705 IC50 = 2120 nM T06273 C6HE2X 60690891 IC50 = 1122.02 nM T06273 C2L6FN 60792847 IC50 = 5600 nM T06273 C9Z5GM 64246802 IC50 = 9400 nM T06273 C4KTU8 66560845 IC50 = 45 nM T06273 CXFG82 66716626 EC50 = 16000 nM T06273 CSC69U 66716715 IC50 = 29 nM T06273 CNL13I 66716735 EC50 = 15000 nM T06273 CF6Y9Z 66716783 IC50 = 17 nM T06273 CB24VJ 66716800 EC50 = 10 nM T06273 C3ZCW7 66716805 IC50 = 56 nM T06273 CD7UX4 66716807 EC50 = 14000 nM T06273 CPSB37 66716841 IC50 = 18 nM T06273 C78KGH 66716854 EC50 = 20 nM T06273 C1RV2K 66716876 EC50 = 20 nM T06273 CEJK92 66716892 EC50 = 9000 nM T06273 CK38YS 66716901 EC50 = 14000 nM T06273 CNBA40 66716932 EC50 = 20 nM T06273 C1XFL3 66716949 EC50 = 20 nM T06273 CE76PS 66716956 EC50 = 10 nM T06273 CP02BL 66717080 EC50 = 16000 nM T06273 C6VXD8 66717138 EC50 = 9000 nM T06273 C1AZ4O 66717208 EC50 = 18000 nM T06273 C1FWI2 66717219 EC50 = 60 nM T06273 CEM82R 66717273 IC50 = 89 nM T06273 C4B1WA 66801593 IC50 = 100000 nM T06273 CN8AS7 67072266 EC50 = 14 nM T06273 CK4DJ3 67189726 IC50 = 500 nM T06273 C72RUQ 67194320 IC50 = 6600 nM T06273 CD3HT9 67960134 IC50 > 100000 nM T06273 C63NJU 68702840 IC50 = 30 nM T06273 C2JKD9 69004309 IC50 = 180 nM T06273 CRF45T 69319479 Ki = 17 nM T06273 C5ME9L 69319562 Ki = 7 nM T06273 CU1G0T 69319608 Ki = 0.9 nM T06273 C3UFV5 69320408 Ki = 2.5 nM T06273 C4WO6P 69320908 Ki = 1.3 nM T06273 CHV0X6 69323356 Ki = 3.5 nM T06273 C8Z7TR 69323654 Ki = 0.7 nM T06273 CX23CL 69323690 Ki = 1.8 nM T06273 CMI1X7 69323902 Ki = 0.9 nM T06273 C9X6QM 70264189 IC50 = 20 nM T06273 CVRL25 70264499 IC50 = 27 nM T06273 C89ZSL 70265346 IC50 = 94 nM T06273 CLTE73 70690554 Ki = 17 nM T06273 C0SJ2R 70692707 Ki = 0.9 nM T06273 C7QLY3 71464718 IC50 > 10000 nM T06273 C6NUT0 71488522 IC50 = 3.2 nM T06273 CM4Y1G 71543402 IC50 = 58 nM T06273 C24XZF 71576800 IC50 > 10000 nM T06273 CNTP10 71580615 IC50 = 825 nM T06273 C9SLK1 71580616 IC50 = 636 nM T06273 CK7PH8 71580620 IC50 = 528 nM T06273 CA2F5X 71580621 IC50 = 1452 nM T06273 CWUI37 71580720 IC50 = 651 nM T06273 C8NG9W 71580721 IC50 = 938 nM T06273 CD9LC2 71604562 IC50 = 210 nM T06273 CW26AZ 71604563 IC50 = 36 nM T06273 CLJ73U 71604564 IC50 = 33 nM T06273 CT2I8V 71604565 IC50 = 45 nM T06273 C3SD7H 71604566 IC50 = 1.9 nM T06273 C8G2DY 71604716 IC50 = 156000 nM T06273 C7ULT5 71604717 IC50 = 1390 nM T06273 CV7N1K 71604718 IC50 = 387000 nM T06273 CQJO61 71604719 IC50 = 3460 nM T06273 CC4XL1 71604867 IC50 = 86200 nM T06273 C3WET2 71604868 IC50 = 560 nM T06273 CM02LW 71604869 IC50 = 76600 nM T06273 C8LC4B 71604870 IC50 = 83900 nM T06273 CE72DU 71604871 IC50 = 4810 nM T06273 CS8CI7 71604872 IC50 = 570 nM T06273 C1JAE9 71605030 IC50 = 11230 nM T06273 C4D2GP 71605031 IC50 = 86340 nM T06273 CK1CB8 71605032 IC50 = 145750 nM T06273 C3S6RX 71605210 IC50 = 210 nM T06273 C8MHC4 71605390 IC50 = 19 nM T06273 CJLV14 71605391 IC50 > 10000 nM T06273 C0IMV2 71605392 IC50 = 490 nM T06273 CTIY17 71606571 IC50 = 8800 nM T06273 CLA3C6 71606723 IC50 = 9380 nM T06273 CF8RD3 71606724 IC50 = 9350 nM T06273 C6UV1N 71606725 IC50 > 10000 nM T06273 C1UR4Y 71606726 IC50 = 300 nM T06273 CV05OF 71606727 IC50 = 8720 nM T06273 CWJD48 71606728 IC50 = 8890 nM T06273 CZ7RV3 71606885 IC50 = 8960 nM T06273 C18DOT 71606887 IC50 = 1100 nM T06273 C3UN6K 71606888 IC50 = 0.31 nM T06273 CFRU61 71606889 IC50 = 1.8 nM T06273 CI0GU8 71660496 IC50 > 85000 nM T06273 CZ1H8S 71681176 IC50 > 85000 nM T06273 C2RGP3 71681329 IC50 > 85000 nM T06273 CI5E8F 71681330 IC50 > 85000 nM T06273 C8I0SW 71718052 IC50 = 8520 nM T06273 C82YZD 71736278 IC50 = 267 nM T06273 C2B5MQ 71736447 IC50 = 652 nM T06273 CF5M7C 71736755 IC50 = 465 nM T06273 CX3Z6J 71769158 IC50 = 5140 nM T06273 C8KBG7 71769159 IC50 = 490 nM T06273 C8FBR2 71769160 IC50 = 1170 nM T06273 C8TC7M 71769162 IC50 = 330 nM T06273 C9LWO6 71769164 IC50 = 1070 nM T06273 COHW23 71769168 IC50 = 880 nM T06273 CEFN02 71769170 IC50 = 900 nM T06273 C9VRD7 71769288 IC50 = 570 nM T06273 CHE1A6 71769290 IC50 = 5610 nM T06273 CA5B0U 71769292 IC50 = 320 nM T06273 CO96XF 71819164 IC50 > 19000 nM T06273 CMC2J4 72193935 IC50 > 85000 nM T06273 C46DHU 72724967 IC50 > 85000 nM T06273 C5XHF0 72736758 IC50 = 0.74 nM T06273 CL3J2U 73056614 IC50 > 19000 nM T06273 CK67DZ 73293053 IC50 > 19000 nM T06273 CE4PM3 73293055 IC50 > 19000 nM T06273 CU3D9N 73388373 IC50 > 1995.26 nM T06273 CZY9U8 73441896 IC50 > 5011.87 nM T06273 CR1ZG8 73603315 IC50 = 370 nM T06273 C62CBA 73774956 IC50 = 200 nM T06273 CP4Z0Q 73774959 IC50 = 560 nM T06273 C4GNA2 73776796 IC50 = 2250 nM T06273 CSG0L9 73776799 IC50 = 2150 nM T06273 CF3R6L 73776801 IC50 = 5400 nM T06273 C4B3JH 73776939 IC50 = 13400 nM T06273 CA0O6Z 73776942 IC50 = 1000 nM T06273 CVPG93 74983349 IC50 = 1530 nM T06273 CH3AT1 76280996 IC50 = 2000 nM T06273 CE45NT 76308159 IC50 = 17 nM T06273 CD4JK3 76310216 IC50 = 880 nM T06273 CEH4W3 76310217 IC50 = 1120 nM T06273 C3CN4E 76313907 IC50 = 270 nM T06273 CPU67O 76313908 IC50 > 5000 nM T06273 CEG28K 76314091 IC50 = 30.3 nM T06273 CBT0Z1 76317419 IC50 = 410 nM T06273 C4IUW9 76317420 IC50 = 260 nM T06273 C65UHF 76317440 IC50 = 270 nM T06273 CSQ48V 76317441 IC50 = 770 nM T06273 CK9Y0P 76319006 IC50 = 47 nM T06273 C9ARI0 76319007 IC50 = 58 nM T06273 C5DMZ2 76321146 IC50 = 1280 nM T06273 CZ9G8B 76321172 IC50 = 930 nM T06273 C9Y2QR 76321173 IC50 = 630 nM T06273 CF9LI1 76321174 IC50 = 3000 nM T06273 CP4EY3 76324803 IC50 = 2900 nM T06273 CCS95Y 76324804 IC50 = 1560 nM T06273 CP7RT1 76324971 IC50 = 10.8 nM T06273 CL38EP 76324972 IC50 = 6.3 nM T06273 C0CA2M 76328339 IC50 = 600 nM T06273 CEBC57 76328359 IC50 > 5000 nM T06273 C9FBG2 76328542 IC50 = 18.7 nM T06273 CCH24O 76332028 IC50 = 3000 nM T06273 C6LMA7 76332029 IC50 = 2100 nM T06273 C8ADE1 76335634 IC50 = 3760 nM T06273 C7NBA8 76335635 IC50 = 280 nM T06273 CTL8W9 76335636 IC50 = 220 nM T06273 C3JKW9 76335856 IC50 = 25.8 nM T06273 C6J2WC 76335857 IC50 = 22.1 nM T06273 CI1GP2 76683569 IC50 = 0.5 nM T06273 C8IT9R 76684090 IC50 = 5.4 nM T06273 C9VP6T 86276157 IC50 > 10000 nM T06273 CC0K6Y 86298601 IC50 = 44 nM T06273 C8EX1M 86298602 IC50 = 100 nM T06273 CC0Q8P 86298603 IC50 = 79 nM T06273 C0CJ9F 86298604 IC50 = 86 nM T06273 CVB6T5 86298605 IC50 = 29 nM T06273 C73MUH 86298606 IC50 = 83 nM T06273 CFB90O 89519195 IC50 = 123 nM T06273 C3XO5D 89649815 IC50 > 100000 nM T06273 C2NC6M 90644171 IC50 = 8167 nM T06273 C7YD9Q 90644172 IC50 = 231 nM T06273 CF2C3G 90644173 IC50 = 133 nM T06273 CM79VU 90644174 IC50 = 284 nM T06273 CDU7E4 90644175 IC50 = 248 nM T06273 CK6NI0 90644176 IC50 = 119 nM T06273 CVBU61 90644177 IC50 = 830 nM T06273 CWA29S 90644178 IC50 = 860 nM T06273 C2GK6X 90644179 IC50 = 400 nM T06273 C9VB4I 90644180 IC50 > 10000 nM T06273 CFM3L5 90644181 IC50 = 600 nM T06273 C2JFU5 90644182 IC50 = 200 nM T06273 CX9B5E 90644183 IC50 = 1100 nM T06273 C1ZNY5 90644184 IC50 = 300 nM T06273 CZ9O8K 90644185 IC50 = 100 nM T06273 CB5CT1 90644186 IC50 = 100 nM T06273 CT4N2O 90644187 IC50 = 100 nM T06273 C3GQ0Y 90644188 IC50 > 10000 nM T06273 COF39B 90644189 IC50 = 6429 nM T06273 CKV5Z4 90644190 IC50 = 1673 nM T06273 C74QYS 90644191 IC50 = 10000 nM T06273 C5L8CR 90644820 IC50 > 25000 nM T06273 CJH4S0 90644821 IC50 = 8440 nM T06273 C46LJC 90644822 IC50 = 6340 nM T06273 CZM14K 90644823 IC50 = 10440 nM T06273 CN7P2R 90644824 IC50 > 25000 nM T06273 C8LQZ9 90644825 IC50 > 25000 nM T06273 C7KY4B 90644826 IC50 = 2450 nM T06273 CHAD15 90644827 IC50 = 3620 nM T06273 C16XKW 90644828 IC50 > 25000 nM T06273 C7SZ3F 90644829 IC50 > 25000 nM T06273 CU3VR6 90644830 IC50 = 2430 nM T06273 CN29DX 90644831 IC50 = 16200 nM T06273 CY7Q2W 90644832 IC50 = 389.05 nM T06273 C7AWT3 90644833 IC50 = 4650 nM T06273 C05SBA 90644834 IC50 = 6090 nM T06273 CM43IE 90644835 IC50 = 3620 nM T06273 C9YB4N 90644836 IC50 = 3300 nM T06273 C1Z0KH 90644837 IC50 > 10000 nM T06273 C3VQ0U 90644838 IC50 = 2140 nM T06273 C09BPX 90644839 IC50 = 813 nM T06273 C6OVD0 90644840 IC50 = 531 nM T06273 C6SA5Q 90644841 IC50 = 753 nM T06273 CKVA38 90644842 IC50 > 10000 nM T06273 CZT2M6 90644843 IC50 > 10000 nM T06273 C79ILK 90644844 IC50 > 10000 nM T06273 CIGD78 90644845 IC50 > 10000 nM T06273 C9GXC4 90644846 IC50 = 544 nM T06273 CVD6T2 90644847 IC50 = 2070 nM T06273 CGFX75 90644848 IC50 = 114 nM T06273 C7BS4G 90644849 IC50 = 718 nM T06273 CLMY42 90644850 IC50 = 223 nM T06273 CXU59P 90644851 IC50 = 1210 nM T06273 CL51HM 90644852 IC50 = 176 nM T06273 CTC18Y 90644853 IC50 = 445 nM T06273 CMZ2Q8 90644854 IC50 = 79 nM T06273 CO78KP 90644855 IC50 = 113 nM T06273 C2XR5Q 92045137 IC50 = 1 nM T06273 C0PIC2 101897062 IC50 = 216.2 nM T06273 CV0NZ7 105539834 IC50 = 77000 nM T06273 CLZ1U3 118498201 IC50 = 730 nM T06273 C1VB9L 118507411 IC50 = 1200 nM T06273 CIK60V 118708492 IC50 = 123.6 nM T06273 C9POS1 118708493 IC50 = 78.62 nM T06273 CUI8V5 118708495 IC50 = 94.88 nM T06273 CGFL69 118708499 IC50 = 85.53 nM T06273 C3E0NP 118708502 IC50 = 72.34 nM T06273 C0Q4BA 118708505 IC50 = 39.61 nM T06273 C34XOL 118708506 IC50 = 10.84 nM T06273 CM5LO4 118708509 IC50 = 107.8 nM T06273 C17CMN 118708510 IC50 = 46.12 nM T06273 CJU29X 118726257 IC50 = 1634.7 nM T06273 C0REJ6 118726258 IC50 = 564.8 nM T06273 CE8KJ2 118732814 IC50 > 20000 nM T06273 CT4WJ8 118732815 IC50 > 20000 nM T06273 CBZ17N 118732816 IC50 > 20000 nM T06273 C1NFU5 118732817 IC50 = 8912.51 nM T06273 CN6SH8 118732818 IC50 = 2400 nM T06273 CF5JT3 118732819 IC50 = 7300 nM T06273 C31AGD 118732820 IC50 = 194.98 nM T06273 CCUW14 118732821 IC50 = 10471.29 nM T06273 C5D4AC 118732822 IC50 = 9700 nM T06273 CKP85E 118732823 IC50 = 389.05 nM T06273 CD4Q2E 118732824 IC50 = 588.84 nM T06273 CAP23E 118732825 IC50 = 800 nM T06273 C4OI5V 118732826 IC50 = 4365.16 nM T06273 CL9F2G 118732827 IC50 = 1100 nM T06273 CZIQ71 118732828 IC50 = 700 nM T06273 C8B7LM 118737587 IC50 = 3.8 nM T06273 CB1SC4 118905298 IC50 = 5.8 nM T06273 CG47YS 118905549 IC50 = 3.9 nM T06273 CBTD43 118905796 IC50 = 3.3 nM T06273 C79MTN 121398248 EC50 > 150000 nM T06273 CLZ1D4 121398509 EC50 > 150000 nM T06273 CRIH72 121398630 EC50 > 150000 nM T06273 CRK45H 122177906 IC50 = 257.04 nM T06273 C8GS6E 122177907 IC50 = 223.87 nM T06273 C9SXK6 122177908 IC50 = 110 nM T06273 CVCS41 122177963 IC50 = 28 nM T06273 CDX95C 122177964 IC50 = 40.74 nM T06273 CYWJ91 122177965 IC50 = 194.98 nM T06273 CC5R3U 122182179 IC50 = 10630 nM T06273 C8XLA4 122182181 IC50 = 44000 nM T06273 CX2N6P 122182187 IC50 = 32 nM T06273 C0CIL6 122182188 IC50 = 29 nM T06273 CI5H1S 122182310 IC50 = 12 nM T06273 CAT68V 122182311 IC50 = 17000 nM T06273 C3TGE0 122182312 IC50 = 140 nM T06273 C25RGB 122182313 IC50 = 460 nM T06273 CMS2L7 122182314 IC50 = 16000 nM T06273 CKS81I 122182315 IC50 = 310 nM T06273 C4I7SQ 122182317 IC50 = 49 nM T06273 C90HTM 122182318 IC50 = 61 nM T06273 CK6W8D 122182319 IC50 = 2280 nM T06273 CFG4A1 122182320 IC50 = 720 nM T06273 C78KCO 122182321 IC50 = 84 nM T06273 CCQ20Z 122182322 IC50 = 1720 nM T06273 CG2TM5 122182323 IC50 = 1280 nM T06273 CRW8H4 122182324 IC50 = 980 nM T06273 C2XYV9 122182325 IC50 = 5960 nM T06273 CJ5G3P 122186786 IC50 = 2000 nM T06273 CK21GN 122189850 IC50 = 17000 nM T06273 CZAF83 122190528 IC50 = 2697 nM T06273 CB6O1P 122190530 IC50 = 11292 nM T06273 COY8A4 122190531 IC50 = 249.7 nM T06273 C5WJ3L 122190532 IC50 = 6.643 nM T06273 CM4W0P 122190533 IC50 = 3.501 nM T06273 CO4X9P 122190534 IC50 = 2.416 nM T06273 CJR13V 122190536 IC50 = 137.6 nM T06273 C3KV7H 122190537 IC50 = 465.4 nM T06273 C21ZNF 122190538 IC50 = 35.44 nM T06273 C02SDC 122423373 IC50 < 30 nM T06273 C7JG6L 124037118 IC50 = 42 nM T06273 CC1DZ2 125504876 IC50 = 152 nM T06273 CB3EZ7 127034750 IC50 = 3 nM T06273 CEG9O8 127034751 IC50 = 22.6 nM T06273 CTY14P 127035738 IC50 = 16.9 nM T06273 CT37NF 127035739 IC50 = 17.6 nM T06273 CH26IE 129896919 IC50 = 79 nM T06273 CV06MU 131801402 IC50 > 100000 nM T06273 C6PMI3 132576435 IC50 = 39.8 nM T06273 CGTF97 132576436 IC50 = 467 nM T06273 CLR6F7 132576437 IC50 = 92.6 nM T06273 C1OJM4 132576507 IC50 = 15.04 nM T06273 CRQ0L4 132576509 IC50 = 6.16 nM T06273 CMI36O 132601761 IC50 = 28 nM T06273 CL3Y1J 132601762 IC50 = 19 nM T06273 CMWX76 132601763 IC50 = 20 nM T06273 C34XLO 132601764 IC50 = 11 nM T06273 CV8MW6 132601765 IC50 = 13 nM T06273 CQ54WE 133053541 IC50 = 244 nM T06273 C2KU8C 133107908 IC50 > 100000 nM T06273 CU3T8P 135398502 IC50 = 25000 nM T06273 CD1R6Q 135400456 IC50 = 2863 nM T06273 C5FTY2 135400457 IC50 = 1210 nM T06273 CVZ7R3 135401666 IC50 = 25000 nM T06273 CU65XO 135402273 IC50 = 10980 nM T06273 C9PI7O 135402338 IC50 > 10000 nM T06273 C4WO1N 135402695 IC50 = 18770 nM T06273 C0HQF2 135404247 IC50 > 100000 nM T06273 C95RAN 135405744 IC50 = 6429 nM T06273 C52WQD 135405818 IC50 = 23 nM T06273 C2B4QH 135405830 IC50 = 170 nM T06273 CTR37Z 135408753 IC50 = 9500 nM T06273 C0UY3F 135412869 IC50 = 5650 nM T06273 C6FY0X 135416131 IC50 = 1295 nM T06273 C6DBN7 135417258 IC50 = 1244 nM T06273 CCY9H6 135417291 IC50 = 3105 nM T06273 CXMS63 135417422 IC50 = 14000 nM T06273 C1PE8H 135417609 IC50 > 20000 nM T06273 CBX8Q2 135418473 IC50 = 16 nM T06273 CYX12Z 135418758 IC50 = 25000 nM T06273 C47LAF 135418940 IC50 = 74.1 nM T06273 CMCS05 135420896 IC50 > 100000 nM T06273 CIS9K5 135421564 IC50 > 100000 nM T06273 C0XW1Z 135423306 IC50 = 25 nM T06273 CO27RD 135429916 IC50 = 3190 nM T06273 CM5Q1Z 135430309 IC50 = 2718 nM T06273 CGS38Z 135431625 IC50 = 25 nM T06273 CP5D4L 135436639 IC50 = 66 nM T06273 C53SJL 135438096 IC50 = 1970 nM T06273 C0J7AN 135440318 IC50 = 16 nM T06273 CIN80B 135440349 IC50 = 8.3 nM T06273 CRJ50Y 135443460 IC50 = 12 nM T06273 C4MW7F 135443732 IC50 > 10000 nM T06273 CH14EB 135443955 IC50 > 10000 nM T06273 CB4P9V 135444661 IC50 = 65 nM T06273 C49QCH 135448200 IC50 = 304 nM T06273 C5F9MI 135448220 IC50 = 250 nM T06273 C8XI3K 135448518 IC50 = 1700 nM T06273 CZ9GA7 135449434 IC50 = 6606.93 nM T06273 CA0R7X 135452109 IC50 = 424 nM T06273 CS94IZ 135452280 IC50 > 10000 nM T06273 CUQ2M3 135452442 IC50 = 25000 nM T06273 C5AT2Z 135452533 IC50 = 25000 nM T06273 C8B2WT 135454888 IC50 = 39 nM T06273 CQU5O2 135456680 Ki = 100000 nM T06273 C9H1VA 135456692 IC50 = 1589 nM T06273 C8J2PC 135456762 IC50 > 5000 nM T06273 CV0G9T 135460986 IC50 = 8 nM T06273 C4J0QA 135462119 IC50 = 270 nM T06273 CDN02O 135471234 IC50 = 17 nM T06273 C94REQ 135471300 IC50 = 1320 nM T06273 CA76KE 135476518 IC50 = 6 nM T06273 CD65XK 135476522 IC50 = 1000 nM T06273 C6CAH2 135477773 IC50 = 540 nM T06273 CAU6W0 135478037 IC50 = 25000 nM T06273 COHR95 135478170 IC50 = 18200 nM T06273 CHY9C3 135479130 IC50 > 100000 nM T06273 CHK58M 135480520 IC50 = 9010 nM T06273 C2K7TH 135483671 IC50 = 37 nM T06273 C5M6NU 135486056 IC50 = 504 nM T06273 CF54RK 135486068 IC50 = 1800 nM T06273 CEG4P1 135489151 IC50 = 16 nM T06273 C6TUL4 135489577 IC50 = 25000 nM T06273 CHQ49P 135493261 IC50 = 25 nM T06273 CPH56D 135495119 IC50 = 46 nM T06273 C7Y5GK 135495133 IC50 = 12 nM T06273 C8Z6RJ 135495930 IC50 = 7040 nM T06273 CF9PI0 135496179 IC50 = 71 nM T06273 CNI94P 135496193 IC50 = 26 nM T06273 CX5R9U 135497113 IC50 = 34 nM T06273 C8XC6L 135508445 IC50 = 27 nM T06273 C1QUP7 135511907 IC50 = 25 nM T06273 C16ASP 135512367 IC50 = 300 nM T06273 CAZM21 135512456 IC50 = 2.2 nM T06273 C9NY6P 135512543 IC50 = 8886 nM T06273 CJO81C 135513650 IC50 = 856 nM T06273 C7G6BQ 135513721 IC50 > 100000 nM T06273 CDM28Q 135515514 IC50 = 13 nM T06273 CAB4X2 135518296 IC50 = 23 nM T06273 CUO26C 135519366 IC50 = 74 nM T06273 CLQ12E 135522325 IC50 = 18 nM T06273 CB5DX7 135524896 IC50 > 1000 nM T06273 C75QZC 135529346 IC50 = 131 nM T06273 CZN82Y 135529360 IC50 = 12 nM T06273 C9E6RB 135529703 Ki = 13 nM T06273 C8F1ZW 135530844 IC50 = 300 nM T06273 C4LYK0 135530847 IC50 = 160 nM T06273 CZIL59 135530863 IC50 = 36 nM T06273 CO4UB6 135531195 IC50 = 14 nM T06273 CMQK85 135537658 IC50 = 26 nM T06273 CK31EQ 135546482 Ki = 6 nM T06273 CQ06WL 135566761 IC50 = 2120 nM T06273 CT8NG2 135566762 IC50 = 900 nM T06273 C1L2WD 135566841 IC50 = 140 nM T06273 C8PQM0 135566842 IC50 = 6460 nM T06273 C7N1YX 135566845 IC50 = 3100 nM T06273 C08WVI 135566846 IC50 = 2500 nM T06273 CG06FQ 135566852 IC50 = 142 nM T06273 C4BFY3 135566969 IC50 = 685 nM T06273 C59OUK 135566970 IC50 > 100000 nM T06273 C7K5WL 135566971 IC50 > 10000 nM T06273 CN74FK 135566972 IC50 = 2404 nM T06273 CRY12I 135566973 IC50 = 559 nM T06273 CU2I7X 135567125 IC50 = 8200 nM T06273 C37PTU 135567126 IC50 = 6456.54 nM T06273 CC7D0M 135580999 IC50 = 1390 nM T06273 C6AQ5K 135621700 IC50 = 29.8 nM T06273 CX82GQ 135623998 IC50 = 760 nM T06273 CT1DZ8 135644892 IC50 > 20000 nM T06273 C38XBR 135652704 IC50 > 20000 nM T06273 CPQS23 135659965 IC50 = 1030 nM T06273 COYA14 135670654 IC50 = 450 nM T06273 C5RUF8 135677066 IC50 = 28.5 nM T06273 C26XEV 135689567 IC50 = 4700 nM T06273 C2HWA5 135711277 EC50 = 256 nM T06273 C1G4CE 135741330 IC50 = 11200 nM T06273 C2C7QU 135741891 IC50 > 19000 nM T06273 C4ZGO7 135741892 IC50 = 10500 nM T06273 C3K2FZ 135742245 IC50 = 7500 nM T06273 CNM35B 135742247 IC50 = 2650 nM T06273 CWH5M1 135742274 IC50 = 5310 nM T06273 CRSP51 135742319 IC50 = 25000 nM T06273 CIL7K3 135742498 IC50 = 144 nM T06273 CD3SM4 135743681 IC50 = 2.14 nM T06273 CF18DR 135759796 IC50 = 87.4 nM T06273 CLE25F 135800247 IC50 = 8.7 nM T06273 C4J2GU 135813363 IC50 = 67.1 nM T06273 C4D2BH 135875690 IC50 = 7000 nM T06273 C0B4PI 135875691 IC50 > 10000 nM T06273 C76QZF 135875692 IC50 = 92.7 nM T06273 CJ7B0D 135875693 IC50 = 110.3 nM T06273 CVP53Y 135875694 IC50 = 428.1 nM T06273 C4UHN8 135875695 IC50 = 1841.5 nM T06273 CQE3G4 135875696 IC50 > 10000 nM T06273 C4XI2O 135875697 IC50 = 106 nM T06273 CVW1I5 135875698 IC50 = 148.6 nM T06273 CGR2K6 135875699 IC50 = 519.2 nM T06273 CIV29L 135875700 IC50 > 10000 nM T06273 C4KC6Z 135875701 IC50 > 10000 nM T06273 CK39DF 135875703 IC50 = 6.9 nM T06273 CXR51Q 135875704 IC50 = 9720 nM T06273 C3KWU1 135875705 IC50 > 10000 nM T06273 C4JMX6 135875706 IC50 = 3 nM T06273 CPW1F0 135893474 IC50 = 1500 nM T06273 C19ZFB 135901558 IC50 = 780 nM T06273 C4ODX8 135901559 IC50 = 510 nM T06273 CJSZ29 135903054 IC50 = 110 nM T06273 CS83CJ 135905416 IC50 = 1600 nM T06273 C21TIS 135906991 IC50 > 1000 nM T06273 CN8R6L 135906992 IC50 = 600 nM T06273 C4HO0Z 135906994 IC50 > 1000 nM T06273 CJA7L8 135906999 IC50 = 700 nM T06273 C2J4DN 135907000 IC50 = 500 nM T06273 CV15XL 135907001 IC50 = 500 nM T06273 C5HC3X 135907003 IC50 > 1000 nM T06273 CLD1A7 135907005 IC50 = 200 nM T06273 COJ04G 135907012 IC50 = 100 nM T06273 CPW14L 135907013 IC50 = 200 nM T06273 CDT79Y 135908480 IC50 = 30 nM T06273 C8DZ7G 135908481 IC50 = 10 nM T06273 CT7UO1 135910401 IC50 = 700 nM T06273 C6BJY9 135910407 IC50 = 1100 nM T06273 C78FUG 135910419 IC50 = 70 nM T06273 CX3HE5 135910421 IC50 = 80 nM T06273 CO26EA 135910423 IC50 = 300 nM T06273 CKL15Y 135910433 IC50 = 600 nM T06273 CR4C1L 135910442 IC50 = 30 nM T06273 CYM46L 135910455 IC50 = 100 nM T06273 CA0FW1 135910457 IC50 = 140 nM T06273 C92RZC 135910459 IC50 = 140 nM T06273 CM7FQ3 135924304 IC50 = 9.45 nM T06273 CC1J9U 135924321 IC50 = 22.4 nM T06273 C1G9HE 135924322 IC50 = 136 nM T06273 C5OE8D 135924334 IC50 = 1.46 nM T06273 C9G5UW 135924335 IC50 = 68.9 nM T06273 C74WRF 135924347 IC50 = 22.4 nM T06273 CC8IL7 135924349 IC50 = 2.6 nM T06273 C3BC4S 135925898 IC50 = 1210 nM T06273 C5L7GW 135927942 Ki = 5.2 nM T06273 CCE59P 135927976 Ki = 16 nM T06273 CIBG05 135931723 IC50 = 240 nM T06273 CLEV87 135939584 IC50 = 100 nM T06273 CKE95M 135939586 IC50 = 200 nM T06273 CST65J 135939587 IC50 = 150 nM T06273 CI9OE0 135939590 IC50 = 500 nM T06273 C7ZVQ0 135939654 IC50 > 1000 nM T06273 C0IK1P 135960846 IC50 = 249 nM T06273 CTH52V 135960847 IC50 = 274 nM T06273 CO7TD0 135965878 IC50 > 1000 nM T06273 C1Z8VU 135965881 IC50 = 1000 nM T06273 C4CFV0 135965923 IC50 > 1000 nM T06273 CWG6U0 135965958 IC50 = 90 nM T06273 C7BTR9 135965959 IC50 > 1000 nM T06273 CUO12L 135965961 IC50 = 300 nM T06273 CWI4P0 135965990 IC50 > 1000 nM T06273 C4HJ1D 135966031 IC50 = 500 nM T06273 CZ1L5H 135966032 IC50 = 1400 nM T06273 CJI2P9 135966077 IC50 > 1000 nM T06273 CMBR14 135966078 IC50 = 800 nM T06273 CREM32 135971442 IC50 = 540 nM T06273 CJO9S5 135981165 IC50 = 400 nM T06273 C4FU1C 135998415 IC50 = 2.4 nM T06273 CO1SG9 136000589 IC50 = 13 nM T06273 CH8X0K 136016494 IC50 = 9.931 nM T06273 C3T1VY 136042254 IC50 = 17 nM T06273 C87OZJ 136042326 IC50 = 13210 nM T06273 CM8FP6 136053646 IC50 = 105 nM T06273 C49DAT 136053647 IC50 = 4139 nM T06273 CV6J0U 136053699 IC50 = 12 nM T06273 CQUA62 136056842 IC50 = 3.29 nM T06273 CF5YU7 136056880 IC50 = 2.48 nM T06273 C7N3ZG 136094865 Ki = 370 nM T06273 C34BJQ 136100291 IC50 = 5.6 nM T06273 CI6SX0 136104470 IC50 = 1600 nM T06273 C4MGZ3 136104471 IC50 = 15 nM T06273 CYS3L8 136104472 IC50 = 25 nM T06273 CFH4P5 136104473 IC50 = 46 nM T06273 CNP9U2 136104474 IC50 = 286 nM T06273 CQ0F1D 136104475 IC50 = 435 nM T06273 CZP7W5 136104476 IC50 = 103 nM T06273 CU5FV8 136104477 IC50 = 257 nM T06273 C4O5ZS 136104478 IC50 = 35 nM T06273 CEM51Z 136104479 IC50 = 16 nM T06273 CXN86A 136104480 IC50 = 47 nM T06273 CL59FC 136104481 IC50 = 30 nM T06273 CO9QG5 136123441 IC50 = 200 nM T06273 CL7KW9 136123472 IC50 = 400 nM T06273 CZ51UY 136123473 IC50 > 1000 nM T06273 C92BEC 136123474 IC50 = 500 nM T06273 CZLA54 136123475 IC50 = 1300 nM T06273 CO1DY5 136123476 IC50 = 2500 nM T06273 CS5B7O 136130843 IC50 = 3.09 nM T06273 CPV26I 136130844 IC50 = 2.63 nM T06273 CKN3D1 136130845 IC50 = 2.35 nM T06273 CU8SB3 136140118 IC50 = 2.08 nM T06273 CM17GZ 136169700 IC50 = 7.3 nM T06273 C54NVS 136175126 IC50 = 1800 nM T06273 CVH7R6 136175127 IC50 = 120 nM T06273 CS5PH8 136175128 IC50 = 1900 nM T06273 CV3UL0 136186300 IC50 = 6.1 nM T06273 CF05ZI 136186302 IC50 = 2.14 nM T06273 C83TAV 136186303 IC50 = 5.27 nM T06273 CNBU78 136186308 IC50 = 2.29 nM T06273 CMRQ94 136186309 IC50 = 6.18 nM T06273 CWA20I 136186310 IC50 = 2.63 nM T06273 CE4PR2 136186312 IC50 = 4.02 nM T06273 C0GN9C 136186318 IC50 = 3.63 nM T06273 C9WD8N 136186322 IC50 = 6.29 nM T06273 CY94ZB 136215772 IC50 > 5000 nM T06273 C7JEG1 136215773 IC50 > 5000 nM T06273 CF7O2U 136215774 IC50 > 5000 nM T06273 CFP0V5 136215897 IC50 > 5000 nM T06273 C19ELM 136219321 IC50 > 19000 nM T06273 CB19RP 136227775 IC50 > 10000 nM T06273 CW7JB0 136229577 IC50 = 510 nM T06273 CR7Q4L 136232699 IC50 = 71200 nM T06273 CM4PB2 136236970 IC50 = 349 nM T06273 C50JYC 136236972 IC50 = 1100 nM T06273 C1WG3C 136236974 IC50 = 830 nM T06273 CF1H5N 136236975 IC50 = 1400 nM T06273 CU17IT 136236976 IC50 = 410 nM T06273 C71FDZ 136236977 IC50 = 2300 nM T06273 CCL4D6 136236978 IC50 = 5700 nM T06273 C9WHB4 136236979 IC50 = 3900 nM T06273 C68GON 136236980 IC50 = 370 nM T06273 C18MSY 136236981 IC50 = 710 nM T06273 CF01JX 136236982 IC50 = 512 nM T06273 CYF2I1 136236983 IC50 = 2500 nM T06273 C3ZW8J 136236994 IC50 = 790 nM T06273 CN0J1C 136236995 IC50 = 4300 nM T06273 CHJ8I2 136236997 IC50 = 79 nM T06273 C0LB6W 136236998 IC50 = 60 nM T06273 CVB4D7 136237000 IC50 = 1300 nM T06273 CSB3Y1 136237004 IC50 = 120 nM T06273 CW9H8J 136237302 IC50 = 10400 nM T06273 CV6OL8 136237316 IC50 > 19000 nM T06273 CA60VL 136237359 IC50 > 19000 nM T06273 C6JH2X 136237372 IC50 > 19000 nM T06273 C4DB3K 136237396 IC50 > 19000 nM T06273 CMC15J 136239430 IC50 = 189 nM T06273 C5QH3A 136240284 IC50 = 130 nM T06273 C79YHQ 136240285 EC50 = 865 nM T06273 CWQ68B 136240852 IC50 = 77 nM T06273 C9KA0J 136241424 IC50 = 300 nM T06273 C02ZRL 136241633 IC50 = 56.1 nM T06273 C4H7LJ 136241634 IC50 = 31.9 nM T06273 CH12EL 136241635 IC50 = 190 nM T06273 CEWX52 136244045 IC50 > 19000 nM T06273 CR07BF 136244504 IC50 = 5500 nM T06273 CVGF06 136244542 IC50 = 388 nM T06273 CHSN59 136245073 IC50 = 266 nM T06273 C79TCS 136249352 IC50 = 700 nM T06273 CXD14B 136249371 IC50 = 220 nM T06273 C5K3WU 136254399 IC50 = 1008 nM T06273 C35VUY 136264437 IC50 = 1980 nM T06273 C0D8MZ 136264443 IC50 = 645 nM T06273 C42HES 136264450 IC50 = 130 nM T06273 CS2CF9 136265171 IC50 = 7.35 nM T06273 CT1YK8 136265176 IC50 = 1.95 nM T06273 CBU1H5 136265177 IC50 = 9.59 nM T06273 CUPY84 136268378 IC50 > 20000 nM T06273 CBG1S2 136344736 IC50 = 5.85 nM T06273 C1USO0 136368560 IC50 = 1.87 nM T06273 CF3X4M 136372378 IC50 = 1361 nM T06273 C1BCA5 136385195 IC50 = 2.25 nM T06273 CLCV40 136385211 IC50 = 3.89 nM T06273 CA1BO8 136385214 IC50 = 1.6 nM T06273 CSL20F 136385215 IC50 = 24.5 nM T06273 C8HL1S 136385220 IC50 = 108 nM T06273 C7PI1W 136385224 IC50 = 2.02 nM T06273 CPB4A7 136385260 IC50 = 2.36 nM T06273 CFY64M 136385284 IC50 = 3.65 nM T06273 CJO98H 136385309 IC50 = 1.1 nM T06273 CR1PV5 136385312 IC50 = 17.7 nM T06273 CEO1W4 136385313 IC50 = 2.02 nM T06273 CUB67C 136404917 IC50 = 1000 nM T06273 CWH02F 136491252 IC50 = 130 nM T06273 CF80AR 136491263 IC50 > 100000 nM T06273 C6T9OI 136947736 IC50 = 620 nM T06273 C91WJF 136947741 IC50 = 390 nM T06273 CFS5Z4 136947743 IC50 = 3700 nM T06273 CVM4S9 136947751 IC50 = 630 nM T06273 CSV0D9 137189936 IC50 = 7.62 nM T06273 CPB15H 137238780 IC50 = 1.84 nM T06273 CGD2R8 137238781 IC50 = 2.76 nM T06273 CJOV40 137238782 IC50 = 2.08 nM T06273 CEW0Q1 137238783 IC50 = 2.88 nM T06273 C4J7SH 137238784 IC50 = 3.9 nM T06273 CYXU75 137348704 IC50 = 27 nM T06273 CW5ZQ2 137348705 IC50 = 17 nM T06273 C7Z4OF 137631560 IC50 = 49 nM T06273 C53XBH 137631697 IC50 = 1810 nM T06273 CET70O 137632114 IC50 > 1000 nM T06273 CF8LC7 137632525 IC50 = 220 nM T06273 CZXI62 137632887 IC50 = 1.4 nM T06273 CEP1D3 137633502 IC50 = 232 nM T06273 C7K8BH 137633902 IC50 = 857 nM T06273 C4VZ3D 137634410 IC50 = 116 nM T06273 CLS5G2 137634533 IC50 = 83 nM T06273 C6ISO0 137634746 IC50 = 60 nM T06273 CE21YX 137634803 IC50 = 644 nM T06273 CW0EP3 137634822 IC50 = 382 nM T06273 CW0Y7D 137635921 IC50 = 311 nM T06273 CXRO18 137635956 IC50 = 111 nM T06273 CZMR82 137636259 IC50 = 1560 nM T06273 C0JBC6 137636342 IC50 > 100 nM T06273 CC8W9L 137636361 IC50 > 100 nM T06273 CBV7D0 137636391 IC50 = 5.7 nM T06273 CW2M0P 137636515 IC50 > 100 nM T06273 C20CYD 137637241 IC50 = 101 nM T06273 CS7ZQ8 137637696 IC50 = 851.14 nM T06273 C8I9WP 137637737 IC50 = 64 nM T06273 C06XTC 137638662 IC50 = 70 nM T06273 C0SQ6X 137638776 IC50 = 79 nM T06273 CMD4H7 137638789 IC50 = 199 nM T06273 CSX50Y 137639400 IC50 = 19 nM T06273 CPLK81 137639614 IC50 = 54 nM T06273 C71UPO 137640297 IC50 > 100 nM T06273 C7V2RQ 137640411 IC50 = 275.42 nM T06273 C6FUP9 137640545 IC50 = 968 nM T06273 C9WXQ3 137641323 IC50 = 40 nM T06273 CY1TA0 137641523 IC50 = 81 nM T06273 C9N2TJ 137642258 IC50 = 346 nM T06273 C91BYL 137642335 IC50 = 29 nM T06273 CJE2O1 137642565 IC50 = 562.34 nM T06273 CD1O9L 137642588 IC50 > 100 nM T06273 CRU6P4 137642996 IC50 = 83 nM T06273 C9ZR0C 137643480 IC50 = 92 nM T06273 CX1CO3 137643739 IC50 = 250 nM T06273 C46GFQ 137643877 IC50 = 363.08 nM T06273 C4AHB5 137644168 IC50 = 223 nM T06273 C8ME0L 137644549 IC50 = 80 nM T06273 C03XFD 137645265 IC50 = 37 nM T06273 CEKY28 137645432 IC50 = 868 nM T06273 CR2U1A 137645856 IC50 = 9.9 nM T06273 CY93WQ 137646242 IC50 = 6.2 nM T06273 CM21PL 137646367 IC50 = 1548.82 nM T06273 CT37OZ 137646498 IC50 = 30 nM T06273 C6P8EW 137646632 IC50 = 2.76 nM T06273 CBT29W 137646686 IC50 = 100 nM T06273 CT6DM0 137646713 IC50 = 62 nM T06273 C45VMW 137647016 IC50 = 793 nM T06273 CW9E5P 137647708 IC50 = 13.7 nM T06273 CV1OU3 137648137 IC50 > 100 nM T06273 CF0ZT5 137648174 IC50 = 3.1 nM T06273 C9M2OL 137648285 IC50 = 302 nM T06273 CT04QR 137648314 IC50 = 108 nM T06273 CTE9D2 137649108 IC50 = 343 nM T06273 CFE07K 137649237 IC50 > 100 nM T06273 C9DE5H 137649777 IC50 = 316 nM T06273 CA48SI 137650468 IC50 > 100 nM T06273 CFPV98 137650613 IC50 = 29 nM T06273 CM4X9L 137650820 IC50 > 100 nM T06273 CG0P8H 137650831 IC50 = 510 nM T06273 C5NH9W 137651141 IC50 = 316 nM T06273 CKS6D5 137651361 IC50 = 820 nM T06273 C3VJE9 137651383 IC50 > 100 nM T06273 CRV60J 137651431 IC50 = 17 nM T06273 C6USY9 137651641 IC50 = 12 nM T06273 CW5E8U 137651914 IC50 = 75 nM T06273 CH0TI5 137652048 IC50 = 20.43 nM T06273 C49QJY 137652661 IC50 = 81 nM T06273 CIFV24 137652719 IC50 = 818 nM T06273 CCNM13 137654119 IC50 = 1190 nM T06273 C2N0KD 137654171 IC50 = 15 nM T06273 CHJE98 137654341 IC50 = 1150 nM T06273 C4NJ0D 137654356 IC50 = 15 nM T06273 C1HE8S 137654622 IC50 = 68.15 nM T06273 CGXT37 137654655 IC50 > 100 nM T06273 CC4ON1 137656059 IC50 = 13.3 nM T06273 C4UTR7 137656957 IC50 = 230 nM T06273 C24ROM 137657941 IC50 > 100 nM T06273 C6M7VX 137658605 IC50 = 41 nM T06273 C8ABS0 137658730 IC50 > 100 nM T06273 CFVN90 137658777 IC50 = 7.54 nM T06273 CDI2K5 137659059 IC50 = 708 nM T06273 C7B9ZV 137660079 IC50 = 174 nM T06273 CAH6B8 137660345 IC50 > 100 nM T06273 C72FHM 137660379 IC50 = 800 nM T06273 CS7LW6 137661452 IC50 = 34 nM T06273 CC0BD9 137661641 IC50 = 88 nM T06273 CZO06Q 137661866 IC50 = 740 nM T06273 C4R7VI 137701512 IC50 > 20000 nM T06273 C1XSH7 138594194 IC50 = 18187 nM T06273 C0RST4 138594360 IC50 > 20000 nM T06273 C4K7MW 138594363 IC50 > 20000 nM T06273 C48AGS 138594414 IC50 > 20000 nM T06273 CA49EZ 138594436 IC50 > 20000 nM T06273 C13EVQ 138594498 IC50 > 20000 nM T06273 C4L9XQ 138594506 IC50 > 20000 nM T06273 CWVO67 138594578 IC50 > 20000 nM T06273 CN3U9X 138594667 IC50 > 20000 nM T06273 C9HR2J 138594785 IC50 > 20000 nM T06273 CP4NF9 138594790 IC50 > 20000 nM T06273 CF7ZR5 138594952 IC50 > 20000 nM T06273 CURM89 138594969 IC50 > 20000 nM T06273 C72QVS 138595093 IC50 > 20000 nM T06273 CJW84M 138857416 IC50 = 36 nM T06273 C0QEY5 138857417 IC50 = 26.92 nM T06273 CBHK62 139589431 IC50 = 18310 nM T06273 CYP38D 141341800 IC50 = 39.1 nM T06273 C86UAQ 141341806 IC50 = 25.8 nM T06273 CS9A6F 141341808 IC50 = 29.8 nM T06273 C1FE9P 141420190 IC50 = 8.41 nM T06273 CWT79B 141466120 IC50 = 345 nM T06273 CW60NV 141466122 IC50 = 58 nM T06273 C6RZY8 141466124 IC50 = 20 nM T06273 C84QGZ 141466125 IC50 = 130 nM T06273 CZ2HI3 141466137 IC50 = 153 nM T06273 CV6BY1 141466145 IC50 = 250 nM T06273 C15IXJ 141466149 IC50 = 8 nM T06273 C64AQL 141466151 IC50 = 14 nM T06273 CVS5D0 141466159 IC50 = 25 nM T06273 CQ2S3B 141466167 IC50 = 22 nM T06273 CNTJ87 141466171 IC50 = 55 nM T06273 C1HKF6 141466173 IC50 = 40 nM T06273 CGI3Y5 141466177 IC50 = 18 nM T06273 C2TG0A 141466191 IC50 = 16 nM T06273 C6NM4Q 141466199 IC50 = 42 nM T06273 CXN16I 141466203 IC50 = 123 nM T06273 CBQ94P 141466205 IC50 = 36 nM T06273 C3YQJ1 141466206 IC50 = 27 nM T06273 CR2QP0 141466210 IC50 = 14 nM T06273 C53IRC 141466213 IC50 = 25 nM T06273 CR7WQ2 141466219 IC50 = 51 nM T06273 CN6M5U 141466229 IC50 = 86 nM T06273 CP1NZ6 141466233 IC50 = 90 nM T06273 C7E8DR 141466238 IC50 = 58 nM T06273 CX7PZ5 141639950 IC50 > 100000 nM T06273 CI09BF 141726120 IC50 = 13.3 nM T06273 CQ40IO 141746550 IC50 > 50000 nM T06273 CPV32H 145949176 IC50 = 0.4 nM T06273 CV3B6Z 145949294 IC50 = 3.5 nM T06273 CN4LI1 145949467 IC50 = 55.8 nM T06273 CF27HL 145949586 IC50 = 0.1 nM T06273 C0VTS8 145949791 IC50 = 1140 nM T06273 C6XOY4 145950109 IC50 = 156.7 nM T06273 C5BH8K 145950405 IC50 = 44.3 nM T06273 CBR5H2 145950461 IC50 = 103 nM T06273 C8DCI4 145950751 IC50 = 250 nM T06273 CZSP73 145950752 IC50 = 2.1 nM T06273 CH78VG 145950905 IC50 = 1390 nM T06273 CWX2B0 145951303 IC50 = 1990 nM T06273 CH0K8V 145951521 IC50 = 450 nM T06273 CGI2B0 145951891 IC50 = 1.3 nM T06273 CNI08D 145951913 IC50 = 100 nM T06273 CM1L3B 145951996 IC50 = 7.1 nM T06273 CC8EY9 145952032 IC50 = 129.7 nM T06273 C48AWJ 145952206 IC50 = 1193 nM T06273 C1LO3G 145952286 IC50 = 1118 nM T06273 CC5YZ7 145952328 IC50 = 2.4 nM T06273 CC82NT 145952335 IC50 = 2535 nM T06273 CHZ3B7 145952366 IC50 = 0.9 nM T06273 CNE4R3 145952501 IC50 = 12.6 nM T06273 CAR58U 145952629 IC50 = 112.2 nM T06273 CFOS14 145952683 IC50 = 1237 nM T06273 CXI9H4 145952767 IC50 = 510 nM T06273 CK1O5P 145953164 IC50 = 320 nM T06273 C0J7UP 145953198 IC50 = 1419 nM T06273 CN80UT 145953368 IC50 = 57.1 nM T06273 CI19VJ 145953381 IC50 = 1700 nM T06273 CO16LA 145953485 IC50 = 24.9 nM T06273 C2YG8W 145954095 IC50 = 4.2 nM T06273 CAN19J 145954692 IC50 = 100.1 nM T06273 C35UIB 145954718 IC50 = 2.6 nM T06273 CJ8FG0 145954839 IC50 = 2969 nM T06273 C82KLB 145954883 IC50 = 877 nM T06273 CQR09L 145954904 IC50 = 3881 nM T06273 C1KD9I 145954997 IC50 = 0.6 nM T06273 CCB5G3 145955102 IC50 = 51.4 nM T06273 CYI79M 145955367 IC50 = 70.5 nM T06273 C14RMT 145955534 IC50 = 0.02 nM T06273 C6IV2D 145955549 IC50 = 0.4 nM T06273 CSE1C4 145955681 IC50 = 2.3 nM T06273 CA8IM1 145955710 IC50 = 90 nM T06273 CN1F4V 145956133 IC50 = 2395 nM T06273 C3OMW2 145956187 IC50 = 141.4 nM T06273 C2TAU7 145956224 IC50 = 174.9 nM T06273 CO79AW 145956303 IC50 = 52.2 nM T06273 CHF70V 145956391 IC50 = 11.2 nM T06273 C1QWK9 145956709 IC50 = 109.5 nM T06273 C0S7FE 145956805 IC50 = 5.1 nM T06273 CC2V7H 145956833 IC50 = 130 nM T06273 C3Q6YV 145956975 IC50 = 33.9 nM T06273 CDI4T3 145957012 IC50 = 2586 nM T06273 C7RL9U 145957093 IC50 = 323.7 nM T06273 C56CUT 145957106 IC50 = 526.1 nM T06273 CAES84 145957591 IC50 = 29.1 nM T06273 C0GXD3 145957654 IC50 = 5.4 nM T06273 CP0X4R 145957773 IC50 = 6.1 nM T06273 C5SG1U 145957836 IC50 = 4397 nM T06273 CK67MD 145958069 IC50 = 190 nM T06273 C8UPE5 145958253 IC50 = 32.4 nM T06273 C58VXI 145958732 IC50 = 970 nM T06273 C48XPR 145958999 IC50 = 233.7 nM T06273 C7GMB4 145959173 IC50 = 1.4 nM T06273 COU95V 145959473 IC50 = 224.9 nM T06273 C9WVK7 145959724 IC50 = 36.5 nM T06273 C5SP6G 145959799 IC50 = 65.4 nM T06273 CD0Y8T 145959884 IC50 = 0.2 nM T06273 C57FTQ 145960349 IC50 < 0.1 nM T06273 C26SHY 145960996 IC50 = 96.8 nM T06273 C4R3PL 145962087 IC50 = 140 nM T06273 CLF0O9 145962288 IC50 = 110 nM T06273 CIH79U 145962718 IC50 = 0.5 nM T06273 CV0Y6A 145962719 IC50 = 0.8 nM T06273 CPR0N4 145962722 IC50 > 100000 nM T06273 CUAP78 145963312 IC50 = 83.4 nM T06273 CFA2V6 145963465 IC50 = 19000 nM T06273 CSYU14 145963753 IC50 = 0.9 nM T06273 COT1U7 145964207 IC50 = 25 nM T06273 C5R2FU 145964279 IC50 = 1101 nM T06273 C6B3YK 145964303 IC50 = 1191 nM T06273 CG91DT 145965021 IC50 = 745 nM T06273 C0TBV5 145965137 IC50 = 951 nM T06273 CO1A5L 145965630 IC50 = 51 nM T06273 CLF6R4 145966106 IC50 = 400 nM T06273 C8X6FH 145967058 IC50 = 1263 nM T06273 CVCQ57 145970486 IC50 = 939 nM T06273 CD2VX1 145971228 IC50 = 9.7 nM T06273 CD86CE 145971751 IC50 = 430.9 nM T06273 C6HOA3 145972257 IC50 = 452.8 nM T06273 CQ6X9V 145972326 IC50 = 304 nM T06273 CK5EF2 145972414 IC50 = 3118 nM T06273 C5OVD6 145972651 IC50 = 0.8 nM T06273 CYE30O 145973023 IC50 = 446 nM T06273 C6UH0Q 145973444 IC50 = 47 nM T06273 CNEB04 145973889 IC50 = 99 nM T06273 CWT2P8 145974066 IC50 = 284 nM T06273 CT87LW 145974068 IC50 = 296.6 nM T06273 CA65UC 145974539 IC50 = 1105 nM T06273 CQD4I1 145975136 IC50 = 1055 nM T06273 CIUY49 145975974 IC50 = 551.6 nM T06273 CQF82C 145976829 IC50 = 136 nM T06273 CU5FP4 145977464 IC50 = 2.9 nM T06273 CZ5PN3 145977729 IC50 = 147 nM T06273 CAB5U8 145978449 IC50 = 277 nM T06273 CK96CU 145978567 IC50 = 1255 nM T06273 CDTA25 145980841 IC50 = 25 nM T06273 C19UOE 145981852 IC50 = 92 nM T06273 C6VLE2 145987066 IC50 = 25 nM T06273 C2JN9I 145991734 IC50 = 37 nM T06273 CF01EN 145992009 IC50 = 15 nM T06273 C6RPG0 146014481 IC50 = 6.026 nM T06273 CPY72O 153951026 IC50 = 910 nM T06273 CLKO63 155510989 IC50 = 37.15 nM T06273 CGH08E 155511904 IC50 = 1.096 nM T06273 CG07YP 155512189 IC50 = 0.7244 nM T06273 CKIA71 155512592 IC50 = 58 nM T06273 C8UYW4 155512651 IC50 = 0.6457 nM T06273 C70LFT 155512744 IC50 = 28.84 nM T06273 CK63OT 155513410 IC50 = 2.57 nM T06273 CMZR80 155513562 IC50 = 1.175 nM T06273 CSP2N8 155513692 IC50 = 2400 nM T06273 CA3OQ8 155514140 IC50 > 50 nM T06273 C9RP5U 155516995 Ki = 1.92 nM T06273 C57EUG 155517403 IC50 > 50 nM T06273 CSR58J 155518352 IC50 = 30 nM T06273 CF5J1D 155518525 IC50 = 2220 nM T06273 CI5KF8 155518636 IC50 = 22 nM T06273 C1DL6E 155518640 IC50 > 20000 nM T06273 CV0EF2 155518789 IC50 = 1.122 nM T06273 C4YJ7D 155519722 IC50 = 338000 nM T06273 C7J0XG 155519774 IC50 = 54 nM T06273 C2Z3RJ 155519958 IC50 = 21.8 nM T06273 CQ8IY2 155521429 IC50 = 51 nM T06273 CHV6T4 155521523 IC50 > 20000 nM T06273 CPH4N0 155522032 IC50 = 97 nM T06273 CUI64O 155522393 IC50 = 46.77 nM T06273 CUM52X 155522687 IC50 > 20000 nM T06273 C2LV0R 155522749 IC50 = 5880 nM T06273 C2H1ZX 155523123 IC50 = 66 nM T06273 C92WIK 155523486 IC50 > 50 nM T06273 C4RD3Z 155523548 IC50 = 21 nM T06273 C5YRO7 155523613 IC50 = 58 nM T06273 CT2P6V 155523711 IC50 > 50 nM T06273 CWK3O5 155524058 IC50 = 31.62 nM T06273 CN4EV1 155526203 IC50 = 66 nM T06273 CUP28Y 155526492 IC50 = 110 nM T06273 CV5D1R 155526501 IC50 > 50 nM T06273 CN9H3Q 155526650 IC50 = 8840 nM T06273 CVPN76 155527263 IC50 = 75 nM T06273 CK7CH6 155527948 IC50 = 194.98 nM T06273 CPLV31 155528423 IC50 = 0.8318 nM T06273 C5Z7SQ 155528446 IC50 = 0.4365 nM T06273 CEP6Y5 155528458 IC50 > 20000 nM T06273 CK90DI 155528679 IC50 = 6560 nM T06273 CLR5E0 155529239 IC50 = 52.48 nM T06273 CIUS95 155529820 IC50 = 92 nM T06273 CJ8H2Z 155530382 IC50 > 50 nM T06273 CFHI87 155531235 IC50 = 4860 nM T06273 CH8ST1 155531582 IC50 = 15.49 nM T06273 C09PYD 155532212 IC50 > 20000 nM T06273 C2IL8E 155533692 IC50 = 33.11 nM T06273 CDAO46 155533875 IC50 > 50 nM T06273 CCS7P2 155534031 IC50 > 50 nM T06273 CCR95S 155534656 IC50 = 41.69 nM T06273 CS0O1N 155535359 IC50 = 97 nM T06273 CV2MX1 155535415 IC50 > 20000 nM T06273 CS7YQ1 155535416 IC50 = 15400 nM T06273 CG9X8C 155535594 IC50 = 21.7 nM T06273 CO6BZ1 155535784 IC50 > 50 nM T06273 CPRG27 155536048 Ki = 10.6 nM T06273 CUK02D 155536515 IC50 = 4590 nM T06273 C3BDY5 155536588 IC50 = 112 nM T06273 CPKV96 155536947 IC50 > 50 nM T06273 CY8RJ7 155537249 IC50 = 16.98 nM T06273 C0ESO2 155537391 IC50 > 50 nM T06273 CAQJ06 155537475 IC50 = 97.72 nM T06273 CS65JI 155537679 IC50 = 950 nM T06273 CWM48X 155538013 IC50 > 20000 nM T06273 CVJQ18 155538037 IC50 = 350 nM T06273 CR3B1W 155538039 IC50 > 50 nM T06273 CM94HZ 155539438 IC50 = 4820 nM T06273 CEP29T 155539891 IC50 = 103 nM T06273 CU65VW 155540828 IC50 > 20000 nM T06273 C7W1DJ 155541447 IC50 = 46.77 nM T06273 CYWG48 155541643 IC50 = 29.51 nM T06273 C9VQO8 155541970 IC50 > 50 nM T06273 CJE20U 155543234 IC50 = 0.6918 nM T06273 C9INM1 155543325 IC50 > 20000 nM T06273 CY48WX 155543524 IC50 = 0.6761 nM T06273 C16YUH 155543913 IC50 > 50 nM T06273 C5N9CJ 155544864 IC50 = 1820 nM T06273 CKC5E3 155545037 IC50 > 50 nM T06273 CG0J7F 155545779 IC50 = 3.89 nM T06273 CS0I4N 155546205 IC50 = 6.166 nM T06273 C8FWY4 155549045 IC50 > 50 nM T06273 CO0E8F 155549220 IC50 > 20000 nM T06273 CBR3M2 155549878 IC50 = 75.86 nM T06273 C9B0VO 155549990 IC50 = 38.02 nM T06273 CPJ75W 155551186 Ki = 0.56 nM T06273 C0JEH6 155551208 IC50 = 9.55 nM T06273 CX2SP3 155551741 IC50 = 10 nM T06273 C6H3MX 155551959 IC50 > 50 nM T06273 CWC03X 155552728 IC50 > 50 nM T06273 CY1WI2 155552891 IC50 = 85.11 nM T06273 C4P3QD 155553178 IC50 > 20000 nM T06273 C1IZF4 155553328 IC50 = 20 nM T06273 CJ8XG3 155553738 IC50 = 28 nM T06273 C0CGI2 155554382 IC50 > 50 nM T06273 CVO72Z 155554427 IC50 = 3200 nM T06273 C84KXJ 155555515 IC50 = 1.072 nM T06273 C1TW9S 155555707 IC50 = 7.943 nM T06273 CIYH06 155556919 IC50 > 20000 nM T06273 CQ8OD5 155559030 IC50 > 50 nM T06273 C2C3NG 155559388 IC50 = 8080 nM T06273 C16DHI 155559491 IC50 = 29 nM T06273 CAC89B 155559886 Ki = 1.48 nM T06273 CM48BL 155560098 IC50 > 50 nM T06273 C2A0TH 155560210 IC50 = 1.29 nM T06273 C0EC4U 155561767 IC50 = 57.54 nM T06273 C46UYI 155562058 IC50 > 20000 nM T06273 CVX7E6 155562207 IC50 = 95.5 nM T06273 C0JRI5 155562814 IC50 = 0.8318 nM T06273 CLJ64M 155562830 IC50 = 139 nM T06273 C6G1SQ 155562883 IC50 = 79.43 nM T06273 C42IWG 155563801 IC50 > 50 nM T06273 C9SX6J 155563867 IC50 = 330 nM T06273 CH1YV0 155563874 IC50 > 50 nM T06273 COH6X1 155564702 IC50 > 20000 nM T06273 CSI7Q1 155565373 IC50 = 66 nM T06273 CZK5Q4 155566057 IC50 > 50 nM T06273 CJH14L 155566731 IC50 = 28.18 nM T06273 CK3UF6 155567820 Ki = 41.5 nM T06273 CTW09V 155568616 IC50 = 53.7 nM T06273 CW8F7S 155568824 IC50 = 43.7 nM T06273 C6NY3Z 155569079 IC50 = 4.898 nM T06273 CE03RY 155569264 IC50 = 67.61 nM T06273 C5YWZ4 155569271 IC50 = 28 nM T06273 CM0DA7 44318575 IC50 = 89 nM T06273 D00OZA 25208746 IC50 = 2300 nM T06273 D00RIX 5280443 IC50 = 100000 nM T06273 D00TUB 135471356 IC50 = 289 nM T06273 D00WMC 790259 IC50 = 753 nM T06273 D01EVX 135875707 IC50 = 1200 nM T06273 D01YIR 1511 Ki = 6 nM T06273 D02GPJ 9948440 IC50 = 18 nM T06273 D02MPP 98487 IC50 = 17000 nM T06273 D02QZF 44549372 IC50 = 130 nM T06273 D02XLC 44407565 IC50 = 5000 nM T06273 D03BQJ 688829 IC50 = 7079.46 nM T06273 D03JTS 1720 IC50 = 26 nM T06273 D03VNZ 44407700 IC50 = 750 nM T06273 D04ATU 11736764 IC50 = 300 nM T06273 D04QRM 135566764 IC50 = 6300 nM T06273 D04TDX 25209058 IC50 = 1100 nM T06273 D04UPQ 11288114 EC50 = 95 nM T06273 D04WDX 4858 IC50 = 10.9 nM T06273 D04ZQJ 690181 IC50 = 224 nM T06273 D05GMW 44407566 IC50 = 2000 nM T06273 D05HJG 10130246 IC50 = 540 nM T06273 D05RXG 18369509 IC50 = 410 nM T06273 D05WYN 44403402 IC50 = 119 nM T06273 D05XMG 9797108 Ki = 6.4 nM T06273 D05ZTI 342403 IC50 = 9100 nM T06273 D06NKJ 135439437 IC50 > 10000 nM T06273 D06XVV 64048 IC50 = 8100 nM T06273 D07AGU 150664 IC50 = 1900 nM T06273 D07BBR 25190932 EC50 = 180 nM T06273 D07BPT 135457978 IC50 = 104 nM T06273 D07CRG 10284 IC50 = 9 nM T06273 D07SRJ 135463574 IC50 = 490 nM T06273 D07WPL 2072 IC50 = 940 nM T06273 D08GMO 25218519 IC50 = 87 nM T06273 D08QWR 616651 IC50 = 770 nM T06273 D08XPZ 25208598 IC50 = 3400 nM T06273 D0B2WX 135407310 IC50 = 891 nM T06273 D0E0QT 25190929 IC50 = 500 nM T06273 D0E5EW 135531482 IC50 = 795 nM T06273 D0EI6X 16221809 IC50 = 180 nM T06273 D0F8ZI 44403357 IC50 = 23 nM T06273 D0FF4M 345678 IC50 = 7500 nM T06273 D0G5VD 135492389 IC50 = 105 nM T06273 D0GA0Y 135463623 IC50 = 504 nM T06273 D0GJ8U 44403404 IC50 = 950 nM T06273 D0I2AF 44549505 IC50 = 71 nM T06273 D0IX3I 44549251 IC50 = 24 nM T06273 D0K2PD 1645 Ki = 3100 nM T06273 D0K7JT 25208747 IC50 = 5800 nM T06273 D0L1NQ 25208596 IC50 = 15000 nM T06273 D0L1RZ 9965481 IC50 = 71 nM T06273 D0M6WJ 10535869 IC50 = 116 nM T06273 D0M9TW 25218518 IC50 = 101 nM T06273 D0NU5Z 11506860 IC50 = 40 nM T06273 D0O0GA 25190931 EC50 = 225 nM T06273 D0O6WW 135528341 IC50 = 1034 nM T06273 D0OF1I 135417274 IC50 > 10000 nM T06273 D0PT1K 44549375 IC50 = 24 nM T06273 D0R7HU 18382004 IC50 = 10000 nM T06273 D0S0RK 10680 IC50 = 1380.38 nM T06273 D0S8HZ 21195867 IC50 = 500 nM T06273 D0T5TT 25208905 IC50 = 2200 nM T06273 D0TH7S 44549373 IC50 = 100 nM T06273 D0U5WY 135508369 IC50 = 1100 nM T06273 D0UF0U 25208904 IC50 = 3700 nM T06273 D0VY5O 9925908 EC50 = 3 nM T06273 D0XZ5D 44549374 IC50 = 14 nM T06273 D0Y1MH 135471354 IC50 = 1200 nM T06273 D0YJ3Q 5322065 IC50 = 7500 nM T06273 D0Z3PB 25208752 IC50 = 800 nM T06273 D0Z9DY 44156952 IC50 = 900 nM T78349 D0K8KX 5280343 IC50 = 1400 nM T78349 CVF5M9 66672 IC50 = 44400 nM T78349 CE3XG2 265580 IC50 = 97400 nM T78349 C3X6HM 1801184 IC50 = 6210 nM T78349 C1JAC5 11425923 Ki = 50 nM T78349 CST06N 16746297 Ki = 590 nM T78349 CNE94V 16746321 Ki = 1050 nM T78349 CLK0Y4 16746438 Ki = 350 nM T78349 CB2HG0 16746461 Ki = 800 nM T78349 C0ZR5T 16746465 Ki = 1100 nM T78349 CRQ16E 24868003 Ki = 570 nM T78349 C0SY2T 132251198 Ki > 100 nM T78349 CND52I 132251245 Ki > 100 nM T78349 CTL8B0 132251294 Ki = 56 nM T78349 C3X5RV 132251295 Ki > 200 nM T78349 CAW73S 132251300 Ki > 200 nM T78349 CIL82X 132251303 Ki = 12.8 nM T78349 C9WRL2 132251354 Ki > 300 nM T78349 C1DO0Y 132251374 Ki > 100 nM T78349 C19IUS 137633595 IC50 = 41900 nM T78349 CRU5O2 137633625 Ki > 100 nM T78349 CFE69X 137635149 Ki = 15 nM T78349 C8CP3E 137637060 IC50 = 380 nM T78349 CLR3V5 137638771 Ki > 200 nM T78349 C5H1ZO 137651476 IC50 = 69600 nM T78349 CT68SX 137652621 Ki = 41 nM T78349 C23OIM 137655418 Ki = 81 nM T78349 C7M9CR 137657529 Ki = 55 nM T78349 C2E6US 137657577 Ki > 100 nM T78349 CZWR03 137659568 Ki = 48 nM T24836 D0I0RJ 16231 IC50 > 50000 nM T24836 D0J0BU 10275777 IC50 > 10000 nM T24836 D0M7JT 216210 Ki = 20930 nM T24836 D01MUU 183797 IC50 = 1300 nM T24836 D0ID3W 9911502 IC50 > 20000 nM T24836 D0PK7J 56599309 Ki = 3000 nM T24836 D03QJN 9895762 Ki = 1800 nM T24836 CZP0Y1 204101 Ki = 19700 nM T24836 C2Z0XW 445482 Ki = 5200 nM T24836 C4VX9Y 9803558 IC50 > 10000 nM T24836 C1FIN6 9804775 IC50 > 130 nM T24836 C4OTK6 9805415 IC50 > 10000 nM T24836 C6JIT7 9806444 IC50 > 11000 nM T24836 CAG59M 9808035 Ki = 1200 nM T24836 C2AXV0 9809479 Ki > 76000 nM T24836 CS1DL7 9826716 IC50 > 181000 nM T24836 CB82VS 9827306 IC50 > 11000 nM T24836 C5Z2RH 9848091 IC50 > 11000 nM T24836 CIL85V 9871029 IC50 > 11000 nM T24836 C6ZB3K 9872552 IC50 > 11000 nM T24836 C1M2PU 9892103 IC50 > 11000 nM T24836 C7I5RG 9892392 Ki = 500 nM T24836 C1C3VT 9914538 IC50 > 11000 nM T24836 CC0D5H 9915041 Ki = 4600 nM T24836 CL2NV0 9935925 IC50 > 870 nM T24836 C5KS0R 9936020 IC50 > 11000 nM T24836 C49DRC 9936691 IC50 > 11000 nM T24836 C8F5CW 9937921 Ki = 1800 nM T24836 C8LR4T 9938917 Ki = 48710 nM T24836 C0R4GE 9954812 IC50 = 3700 nM T24836 CM7IF6 9956559 Ki > 20000 nM T24836 C2Y0QV 9959268 IC50 > 10000 nM T24836 CBC2K3 9959749 IC50 > 11000 nM T24836 CFQV59 10007890 IC50 > 10000 nM T24836 CF1V4K 10027758 Ki > 18000 nM T24836 CQP65H 10095093 Ki = 180000 nM T24836 C3OG5U 10095865 IC50 > 25100 nM T24836 CW4RZ5 10116936 IC50 > 450 nM T24836 C7PC2K 10185292 IC50 > 170 nM T24836 CO51ZR 10205659 IC50 > 10000 nM T24836 C4Z1LU 10255253 Ki > 18000 nM T24836 C9IAO4 10256095 IC50 = 100 nM T24836 CQ9ZO1 10275412 Ki > 38000 nM T24836 CV10CU 10297977 IC50 > 10000 nM T24836 C1AP6H 10298858 IC50 > 10000 nM T24836 CK9J7X 10343728 IC50 > 25100 nM T24836 C4JC7H 10367232 IC50 = 800 nM T24836 CMNP39 10389039 IC50 > 10000 nM T24836 CLK08Z 10391999 IC50 > 10000 nM T24836 C6AZ8B 10435038 Ki = 43000 nM T24836 CCP2N8 10480374 Ki > 18000 nM T24836 CV0X6G 10480463 IC50 > 11000 nM T24836 CEI65Z 10483775 Ki = 73 nM T24836 CU8N3V 10578280 Ki = 13500 nM T24836 C8SUZ9 10624948 Ki = 48000 nM T24836 CEJ14F 10624997 Ki = 10300 nM T24836 CR5EX8 10648196 Ki = 29000 nM T24836 CPWH69 10648370 Ki = 94000 nM T24836 C5VB1U 10695159 Ki > 1000000 nM T24836 CGYR23 10696955 Ki = 12000 nM T24836 CPGV87 10718240 Ki = 180000 nM T24836 CKOQ35 10767421 Ki > 1000000 nM T24836 C3IN8W 10815545 Ki = 39000 nM T24836 CVQE76 10816339 Ki = 15200 nM T24836 CRDU42 11271947 Ki > 33000 nM T24836 CVI82D 11479420 Ki = 28000 nM T24836 C8GJO7 11754872 IC50 > 33000 nM T24836 CNPW05 11755188 IC50 > 10000 nM T24836 CNO67W 11798089 Ki = 80000 nM T24836 CC6M2W 11849330 IC50 > 33000 nM T24836 C1T6CS 11849331 IC50 > 33000 nM T24836 CRT0N2 11849332 IC50 = 9080 nM T24836 C21OSF 11849333 IC50 = 2040 nM T24836 CLH9U6 11849334 IC50 = 3830 nM T24836 CGB6W0 11849371 IC50 = 750 nM T24836 CX5BV1 11849373 IC50 = 11250 nM T24836 CH7BM8 11849374 IC50 = 44000 nM T24836 C0K7UZ 11849375 IC50 = 53000 nM T24836 CPR12Z 11849376 IC50 = 10910 nM T24836 C82FJL 11849424 IC50 = 1070 nM T24836 C89XNT 11849425 IC50 = 1700 nM T24836 C8TVZ9 11849426 IC50 = 250 nM T24836 CF7UX3 11849427 IC50 = 9280 nM T24836 CW1QF2 11849428 IC50 = 430 nM T24836 CEO7G0 11849429 IC50 = 12650 nM T24836 CR5H3J 11849462 IC50 = 350 nM T24836 C1JBR8 11849463 IC50 = 710 nM T24836 C83JRC 11849464 IC50 > 33000 nM T24836 C19ARJ 15984063 Ki > 150000 nM T24836 CA8Y1K 16046152 Ki = 19000 nM T24836 CNBJ60 16046153 Ki > 76000 nM T24836 C53YRO 16098910 IC50 = 20700 nM T24836 C29WYS 18675086 IC50 = 23000 nM T24836 CB0IQ4 18727607 IC50 > 11000 nM T24836 C31ZAL 18727831 IC50 > 11000 nM T24836 CJY67O 18727833 IC50 > 11000 nM T24836 C02HEA 18727834 IC50 > 11000 nM T24836 CJSL38 18727836 IC50 > 11000 nM T24836 C8AMY9 18727838 IC50 > 11000 nM T24836 CY8AC3 18727841 IC50 > 11000 nM T24836 CD02TK 18727852 IC50 > 11000 nM T24836 C1JMX5 18727855 IC50 > 11000 nM T24836 CO2JG4 20595081 IC50 > 11000 nM T24836 CM7BH1 20595091 IC50 > 11000 nM T24836 CCH5N1 20595225 IC50 > 11000 nM T24836 C2ID8R 20595260 IC50 > 10000 nM T24836 CMT46A 20595328 IC50 > 10000 nM T24836 C7LHE8 20641745 IC50 > 180000 nM T24836 CZ6KH9 20760195 Ki > 76000 nM T24836 CNTI15 21366511 IC50 > 11000 nM T24836 C5S8ZW 21366513 IC50 > 11000 nM T24836 C67QCO 21366574 IC50 > 11000 nM T24836 CS2L1Y 21366575 IC50 > 11000 nM T24836 CX1WM9 21366579 IC50 > 11000 nM T24836 CI0SJ2 21967345 Ki = 9500 nM T24836 CA3N9L 22883564 Ki > 18000 nM T24836 C1R0UD 22883585 Ki = 12000 nM T24836 C13-JAN 22883594 Ki = 4200 nM T24836 CCRD27 23646312 Ki > 37000 nM T24836 C1WE6B 23646315 Ki > 20000 nM T24836 CKH4O5 24180463 Ki > 21000 nM T24836 CJSO87 24849206 Ki > 33000 nM T24836 CN0ZW3 24999867 Ki > 1000 nM T24836 CEM32W 25001205 Ki > 1000 nM T24836 CI8HE3 25138142 IC50 > 33000 nM T24836 C2H4PJ 25166809 Ki > 64000 nM T24836 CKM7Y8 25269170 Ki > 20000 nM T24836 CL7NY5 44274017 IC50 > 10000 nM T24836 CMG90C 44274089 IC50 > 10000 nM T24836 CZRH12 44290033 IC50 > 11000 nM T24836 CUY95P 44290108 IC50 > 11000 nM T24836 C8APX2 44290947 Ki > 18500 nM T24836 CSM3B6 44330879 IC50 = 6560 nM T24836 CE69GW 44331194 IC50 = 73000 nM T24836 CRT4G3 44335601 Ki = 33000 nM T24836 C7Z9WL 44335624 Ki = 180000 nM T24836 C34XTM 44375987 IC50 = 6000 nM T24836 CD0W7C 44376100 IC50 > 180000 nM T24836 C0Y8QD 44376252 IC50 = 170000 nM T24836 C5R2PM 44376328 IC50 = 169000 nM T24836 C5VDG0 44376417 IC50 > 180000 nM T24836 CG64YQ 44376426 IC50 > 180000 nM T24836 C9SD3E 44383242 Ki > 18000 nM T24836 C43KTU 44383519 Ki > 18000 nM T24836 CG7LT1 44385488 IC50 > 11000 nM T24836 C94GZU 44385541 IC50 > 11000 nM T24836 C3T9XK 44385607 IC50 > 11000 nM T24836 CKY0P4 44385611 IC50 > 11000 nM T24836 CUS20V 44385673 IC50 > 11000 nM T24836 CZ8XL6 44385679 IC50 > 11000 nM T24836 CL5BA4 44385729 IC50 > 11000 nM T24836 C3DSN7 44385768 IC50 > 11000 nM T24836 C8USN9 44385769 IC50 > 11000 nM T24836 C2E8DS 44385771 IC50 > 11000 nM T24836 C2VFC6 44385772 IC50 > 11000 nM T24836 CN8V0W 44385779 IC50 > 11000 nM T24836 CBEA65 44385842 IC50 > 11000 nM T24836 CC9M7E 44385869 IC50 > 11000 nM T24836 C8WK4A 44385891 IC50 > 11000 nM T24836 C3D2CL 44385935 IC50 > 11000 nM T24836 CW08OY 44385998 IC50 > 11000 nM T24836 CV6KG4 44386059 IC50 > 11000 nM T24836 CGU69V 44386179 IC50 > 11000 nM T24836 CS65LH 44386185 IC50 > 11000 nM T24836 CU0P5T 44386242 IC50 > 11000 nM T24836 CU9J0D 44386250 IC50 > 11000 nM T24836 C9G7QW 44386322 IC50 > 11000 nM T24836 C31CUG 44386326 IC50 > 11000 nM T24836 C2WCE4 44386371 IC50 > 11000 nM T24836 C52POK 44386417 IC50 > 11000 nM T24836 CRX1I9 44386418 IC50 > 11000 nM T24836 CIBD76 44386484 IC50 > 11000 nM T24836 C8ME4O 44386493 IC50 > 11000 nM T24836 CD4AH3 44386540 IC50 > 11000 nM T24836 CHAO48 44386542 IC50 > 11000 nM T24836 CLNO15 44386637 IC50 > 11000 nM T24836 C81IMH 44386642 IC50 > 11000 nM T24836 C4JB0M 44386841 IC50 > 11000 nM T24836 C5MR1F 44386934 IC50 > 11000 nM T24836 CA45DZ 44387044 IC50 > 11000 nM T24836 C39LUW 44387104 IC50 > 11000 nM T24836 C2QD1K 44387206 IC50 > 11000 nM T24836 C3BX5Y 44412781 Ki > 150000 nM T24836 CO6Z9S 44415089 IC50 = 1120 nM T24836 CR16BF 44434808 Ki > 21000 nM T24836 CQIX73 44434809 Ki > 21000 nM T24836 C5R8HJ 44434815 Ki > 21000 nM T24836 COG34X 44434818 Ki > 21000 nM T24836 C9T1DP 44434835 Ki > 21000 nM T24836 CLOY62 49864459 Ki > 33000 nM T24836 CR8JK9 49864483 Ki > 33000 nM T24836 CVDF05 50908868 IC50 = 395300 nM T24836 CVD91F 50908869 IC50 = 284100 nM T24836 CV8I3U 52942903 IC50 = 103500 nM T24836 C1LEN7 52948297 IC50 = 144500 nM T24836 CA6GQ5 53341037 Ki > 21500 nM T24836 CIKQ81 53345652 Ki > 130 nM T24836 CXWS90 53345968 Ki > 1000 nM T24836 CV60BK 53488415 Ki = 22500 nM T24836 C17MSO 56640092 Ki = 564 nM T24836 CGP7Y6 56640160 Ki = 48 nM T24836 C30AJK 56640226 Ki = 4586 nM T24836 CH1EI8 56954620 Ki = 5.1 nM T24836 C4EHU8 56954732 Ki = 12000 nM T24836 C5C8XO 56954733 Ki = 3510 nM T24836 CST4F0 56954834 Ki = 223 nM T24836 CRK92A 56954952 Ki = 8390 nM T24836 CTE30K 57842560 Ki = 14000 nM T24836 C0C6UB 57842624 Ki = 1800 nM T24836 C7XY5A 57842673 Ki = 2800 nM T24836 C41NSR 57842812 Ki = 41 nM T24836 C9XW1C 57842830 Ki > 10000 nM T24836 CWF0C3 57842850 Ki = 1300 nM T24836 C73CPB 57842913 Ki = 830 nM T24836 C60HCV 57976401 Ki > 21500 nM T24836 CHB27Y 57976410 Ki > 30220 nM T24836 CSC0L5 59020200 Ki > 37600 nM T24836 CPW2H7 59315536 Ki > 10000 nM T24836 CO38AC 59402011 Ki > 64000 nM T24836 CE5A7B 60162406 Ki > 25000 nM T24836 CWOD93 66744646 Ki > 21500 nM T24836 C0SDB3 68020667 Ki > 10000 nM T24836 C6AU1R 70252985 Ki = 68000 nM T24836 CTO5I6 70253788 Ki > 64400 nM T24836 C8A7ZJ 70306716 Ki = 0.46 nM T24836 C4IFW3 70683249 Ki = 0.61 nM T24836 CN38UY 70687492 Ki = 90 nM T24836 C9EL3C 71260387 Ki > 21500 nM T24836 C45SHM 71451304 Ki > 20000 nM T24836 CJPF90 71548883 Ki > 21000 nM T24836 C30ZKJ 71561420 Ki > 15000 nM T24836 CH32TL 71561557 Ki = 3900 nM T24836 C8RW7E 71562631 Ki = 39 nM T24836 C4UHB2 71562760 Ki = 420 nM T24836 C0EM6D 71562761 Ki = 880 nM T24836 CNS21T 71562882 Ki = 3800 nM T24836 C3SBE2 71562883 Ki = 7800 nM T24836 C2NY0B 71563006 Ki > 20000 nM T24836 CG46AZ 71563007 Ki = 4800 nM T24836 C2O4SB 71563124 Ki > 10000 nM T24836 C4CT8O 71563125 Ki = 1600 nM T24836 C78DJQ 71711730 IC50 < 10000 nM T24836 CQ3K2V 71719191 Ki = 4100 nM T24836 CXM6C2 72550813 Ki = 70 nM T24836 CLI36U 72551247 Ki = 190 nM T24836 CFH7S6 76310670 Ki = 400 nM T24836 CUZM48 76314299 Ki = 800 nM T24836 CS92KW 76317870 IC50 > 44000 nM T24836 C9C4BV 76317871 Ki = 300 nM T24836 CWH27L 76317872 Ki = 500 nM T24836 C3BG6X 76321582 Ki = 300 nM T24836 CSY7X9 76325187 Ki = 900 nM T24836 COBF15 76325188 Ki = 300 nM T24836 CO28RN 76325189 Ki = 100 nM T24836 CQ98SD 76325190 Ki = 1600 nM T24836 C9O1BS 76328752 IC50 > 44000 nM T24836 CO3H5T 76328753 Ki = 900 nM T24836 C1I2WQ 76328754 Ki = 200 nM T24836 C59GFM 76328756 Ki = 100 nM T24836 C6CW8M 76332426 Ki = 300 nM T24836 C0BXZ8 76332427 Ki = 1100 nM T24836 CIN46O 86343959 Ki = 1200 nM T24836 CWS28P 86344699 Ki = 39 nM T24836 CMD5V7 86583041 Ki > 21400 nM T24836 CO6U9I 88582319 Ki > 64400 nM T24836 C65TLW 101862198 Ki > 1000000 nM T24836 C28PCL 117749867 Ki = 5700 nM T24836 CHQ5P7 118987013 Ki > 30220 nM T24836 C3YVQ8 122164611 Ki = 725 nM T24836 CY1S5D 122164612 Ki = 155 nM T24836 CK0W2P 127027635 Ki > 60000 nM T24836 CPC0M8 127031390 Ki > 30220 nM T24836 C1BWV2 127035672 Ki > 1000000 nM T24836 CVRY56 127036086 Ki > 1000000 nM T24836 C9B6LT 127037264 Ki > 1000000 nM T24836 C60HLK 127037469 Ki > 1000000 nM T24836 CC7UO1 134133660 Ki = 1600 nM T24836 C9UZI0 134148669 Ki = 220 nM T24836 CR6V9U 134150310 Ki = 175 nM T24836 CG9UL4 134156593 Ki = 340 nM T24836 C6HTD5 135393470 IC50 > 50000 nM T24836 C7NA6E 135393474 IC50 > 50000 nM T24836 CD53CZ 135404951 Ki ~ 18500 nM T24836 C9KLD3 135455964 Ki = 18000 nM T24836 CJWC64 135462427 Ki = 1970 nM T24836 C91UXW 135802775 Ki = 15000 nM T24836 CYQ70K 136053621 IC50 > 11000 nM T24836 CPK6X2 136198635 Ki = 11000 nM T24836 CRJ5S4 136198636 Ki = 5500 nM T24836 C7WE2G 136198637 Ki = 8000 nM T24836 C12UWY 136198638 Ki > 18000 nM T24836 CDQ62V 137637214 Ki > 50000 nM T24836 C2K8JV 137639385 Ki > 50000 nM T24836 CNX46H 137654508 Ki > 50000 nM T24836 CO51HN 139030452 IC50 > 50000 nM T24836 CX07YE 139592452 Ki > 7160 nM T24836 CE6C0A 145970642 Ki = 16300 nM T24836 C4HLX8 146029523 IC50 > 50000 nM T24836 CH59QO 155510375 Ki > 100000 nM T24836 CA81QV 155512709 Ki = 32000 nM T24836 C2VX3G 155512946 Ki > 21500 nM T24836 CG9H4N 155515624 Ki = 130400 nM T24836 C7ZM4R 155515728 Ki = 28017 nM T24836 CFRS54 155516565 Ki = 49340 nM T24836 C1ZSV0 155517054 Ki = 47050 nM T24836 CH0N9A 155523885 Ki > 30000 nM T24836 CYL8M0 155526377 Ki = 93400 nM T24836 CX7CO2 155527010 Ki = 17000 nM T24836 C46AZL 155530642 Ki > 25000 nM T24836 CP8K2J 155531811 Ki = 39740 nM T24836 C0UR8Q 155531991 Ki = 74700 nM T24836 CIHM01 155535907 Ki > 100000 nM T24836 C7JMK4 155538439 Ki > 13000 nM T24836 C9QE5N 155538514 Ki = 62910 nM T24836 CRT3D4 155540148 Ki = 51490 nM T24836 C4CHR9 155542229 Ki = 96500 nM T24836 C4P2GV 155543617 Ki > 25000 nM T24836 CSI5J1 155548907 Ki = 212000 nM T24836 CA5VG2 155552651 Ki = 106100 nM T24836 C5S6HO 155553129 Ki = 46500 nM T24836 C5TV4J 155554082 Ki = 42018 nM T24836 CU8LR3 155555208 Ki > 25000 nM T24836 CXL5D4 155558368 Ki > 100000 nM T24836 C3SXY1 155561904 Ki = 85870 nM T24836 CX5O7K 155562968 Ki > 30000 nM T24836 CK0EA2 155568484 Ki = 4280 nM T24836 D00KJP 10322586 Ki = 2400 nM T24836 D02YIW 1794 IC50 > 50000 nM T24836 D06HOI 44249821 Ki > 18000 nM T24836 D0J1QT 44473100 Ki > 18000 nM T24836 D0JU9N 6914623 Ki > 2800 nM T24836 D0MQ6K 10574241 Ki = 7000 nM T24836 D0ON2Z 204102 Ki > 2300 nM T24836 D0V7TH 76328755 Ki = 40 nM T24836 D0Y5IQ 44255320 IC50 = 50000 nM T89213 D0LI1C 44469321 IC50 > 10000 nM T89213 D0Q3UL 9820766 Ki = 48 nM T89213 D0V2GT 5311023 Ki = 1 nM T89213 CT6RA0 2317 Ki = 1800 nM T89213 C9NG4X 16033 EC50 = 0.03981 nM T89213 C74KDN 624746 IC50 > 10000 nM T89213 C1Q4WZ 1294837 Ki > 6309.57 nM T89213 CF20QJ 4527770 Ki > 31622.78 nM T89213 C39UDN 5312114 IC50 = 8370 nM T89213 CI26VT 9799669 IC50 > 30000 nM T89213 C5MC8Y 9802119 IC50 > 10000 nM T89213 C7DCV0 9805674 Ki = 8 nM T89213 CJ2KX8 9806472 Ki = 5546 nM T89213 CJC47U 9806521 Ki = 7.3 nM T89213 C2GV5J 9807379 Ki = 5.1 nM T89213 CK7QY8 9867212 IC50 > 30000 nM T89213 CG3FU8 9868731 Ki = 29 nM T89213 CT7S5I 9869041 Ki = 1 nM T89213 C0EGK5 9869458 Ki > 10000 nM T89213 C8J2EG 9869677 Ki = 3 nM T89213 CXJL03 9885994 IC50 > 10000 nM T89213 CPGD84 9887225 IC50 > 10000 nM T89213 C2EI3N 9894291 IC50 = 120 nM T89213 CZ31PQ 9908496 Ki = 21 nM T89213 C0A6OH 9911304 Ki = 383 nM T89213 CS92LR 9916525 Ki = 0.75 nM T89213 CWP3V6 9930778 IC50 >> 1000 nM T89213 CA9CQ2 9931301 IC50 = 39 nM T89213 C4QWK3 9932616 Ki = 7 nM T89213 C7NOZ8 9956814 Ki = 5 nM T89213 CJ6BV9 9959777 IC50 = 1.4 nM T89213 CC05RX 9982218 Ki = 16032 nM T89213 C56JMF 9987422 Ki = 0.052 nM T89213 C72HXY 10005032 IC50 > 10000 nM T89213 CH1Q6E 10008757 Ki = 0.037 nM T89213 CK3W5X 10030299 Ki = 0.06 nM T89213 C73QBA 10047509 IC50 > 10000 nM T89213 CUFC30 10051692 IC50 > 10000 nM T89213 C8IVM5 10053818 IC50 = 4.4 nM T89213 C82VAF 10071200 IC50 > 10000 nM T89213 CG2V1H 10076108 Ki = 4.5 nM T89213 CL96TH 10110741 IC50 > 10000 nM T89213 C6IXU4 10293988 Ki > 10000 nM T89213 C8L7WY 10295464 IC50 > 30000 nM T89213 C3M1ON 10326097 Ki = 0.75 nM T89213 CYR59E 10414488 Ki = 1.7 nM T89213 CA1C6E 10418848 Ki = 5 nM T89213 C4HMY5 10429613 IC50 > 10000 nM T89213 CNR16C 10457755 IC50 > 10000 nM T89213 CK6JQ5 10458754 Ki = 15 nM T89213 CB07JL 10472655 Ki = 282 nM T89213 C7M3GI 10505296 Ki = 160 nM T89213 CUS60F 10505977 Ki > 10000 nM T89213 C9F7WZ 10509290 Ki = 17 nM T89213 C84MSG 10524003 Ki = 4.6 nM T89213 CTAE67 10529375 Ki = 140 nM T89213 C0YNJ2 10531064 Ki = 780 nM T89213 CKQ2G1 10531484 Ki = 1.4 nM T89213 CBO13L 10552512 Ki > 10000 nM T89213 C3ARF7 10552954 Ki = 450 nM T89213 C3WHI0 10554007 Ki = 86 nM T89213 CD7T9M 10554097 Ki = 26 nM T89213 C17LZS 10554549 Ki = 65 nM T89213 CQ1P5I 10554658 Ki = 98 nM T89213 C5R0VU 10554910 Ki = 610 nM T89213 C0F9SD 10555187 Ki = 1.9 nM T89213 C4KJR6 10577766 Ki = 80 nM T89213 CO3I6A 10577912 Ki = 100 nM T89213 CX2I4Y 10577995 Ki = 18 nM T89213 CXK54C 10578417 Ki = 690 nM T89213 CIBL17 10599930 Ki = 7300 nM T89213 CCW87K 10600984 Ki = 240 nM T89213 C3I1TZ 10601025 Ki = 470 nM T89213 C2E5LH 10601376 Ki = 700 nM T89213 CL0MH6 10601378 Ki = 980 nM T89213 CYH17Z 10601584 Ki = 7.6 nM T89213 CQH95Z 10601682 Ki = 5500 nM T89213 CSBY18 10605125 Ki = 16 nM T89213 CN3J1U 10605127 Ki = 30 nM T89213 C0FP2G 10619067 Ki = 2310 nM T89213 CO2V3H 10624729 Ki = 3800 nM T89213 CM54NH 10624769 Ki = 43 nM T89213 CAIW12 10624998 Ki = 150 nM T89213 CZ0U1P 10625004 Ki = 440 nM T89213 CUNV20 10625155 Ki = 15 nM T89213 CNY64H 10625178 Ki = 56 nM T89213 CK9IR7 10625207 Ki = 200 nM T89213 CTQ3J4 10625562 Ki = 97 nM T89213 CWP0E7 10625797 Ki > 10000 nM T89213 CZG82Q 10625949 Ki = 17 nM T89213 C0W8MS 10626335 Ki = 18 nM T89213 CG16HR 10647548 Ki > 10 nM T89213 CL41PE 10649770 Ki = 7.8 nM T89213 CIB4C0 10649777 Ki = 17 nM T89213 CZJ2Q9 10649849 Ki = 66 nM T89213 C3L6TA 10671331 Ki = 559 nM T89213 C7MC2O 10672357 Ki = 26 nM T89213 CU8L6M 10673317 Ki = 400 nM T89213 C0MK1J 10673757 Ki = 28 nM T89213 C9JL3S 10673787 Ki = 88 nM T89213 CFG3T2 10674056 Ki = 24 nM T89213 CY07DC 10676562 Ki = 27 nM T89213 C6HQ1X 10692519 Ki = 1260 nM T89213 CU91GE 10696695 Ki = 1400 nM T89213 C0OM9F 10696766 Ki = 82 nM T89213 CDSM69 10700181 Ki = 29 nM T89213 C5X1IF 10718106 Ki > 10000 nM T89213 CXO0H2 10719643 Ki = 7860 nM T89213 C29DNK 10720174 Ki = 75 nM T89213 CBN6P2 10720203 Ki = 1200 nM T89213 C4FAW1 10722606 Ki = 43 nM T89213 CJ9W1K 10741628 Ki = 7000 nM T89213 C1HLC4 10743445 Ki = 910 nM T89213 CGJT78 10744091 Ki = 29 nM T89213 C23QDW 10744510 Ki > 10000 nM T89213 C0VQ6R 10744516 Ki = 71 nM T89213 CP3C6M 10747569 Ki = 7 nM T89213 C6P2QS 10747659 Ki = 6 nM T89213 C7MFL8 10767712 Ki = 2.9 nM T89213 CIZ4O3 10768322 Ki = 7.8 nM T89213 C8X3TS 10768834 Ki = 7.8 nM T89213 C3MT6O 10768859 Ki = 36 nM T89213 CT72CY 10786219 Ki = 7020 nM T89213 CU28XN 10787168 Ki > 10000 nM T89213 C6BW3A 10791009 Ki = 940 nM T89213 CZ43JL 10791454 Ki = 3230 nM T89213 CYB59I 10795082 Ki = 18 nM T89213 CD23YC 10809141 Ki > 100000 nM T89213 C85IKP 10815247 Ki = 4100 nM T89213 C56RAU 10815605 Ki = 1210 nM T89213 C1RGA9 10816198 Ki = 56 nM T89213 C0T5NV 10816575 Ki = 25 nM T89213 C4C2TQ 10818866 Ki = 41 nM T89213 CS4JF0 10820168 Ki = 34.8 nM T89213 CEH6O1 10820196 Ki = 25.7 nM T89213 CD5KW2 10838640 Ki = 690 nM T89213 C3HQD1 10838641 Ki = 83 nM T89213 CO4IB3 10839510 Ki > 10000 nM T89213 CLM2C1 10839529 Ki = 5300 nM T89213 C6B8YE 10842778 Ki = 152 nM T89213 CGT23W 10872843 IC50 > 10000 nM T89213 CFHD79 10915843 IC50 > 10000 nM T89213 CDMB60 10916418 IC50 > 10000 nM T89213 C21PAY 10927348 IC50 > 10000 nM T89213 CJ0OF1 10949261 IC50 > 10000 nM T89213 CM54HE 10959710 IC50 > 10000 nM T89213 C08VWM 10971892 IC50 > 10000 nM T89213 CO98AV 10982716 IC50 > 10000 nM T89213 CI6W3N 10993145 IC50 > 10000 nM T89213 CGSF91 11013840 IC50 > 10000 nM T89213 C1ICL8 11025578 IC50 > 10000 nM T89213 C4UPT2 11057893 IC50 > 10000 nM T89213 CKC6D3 11133371 IC50 > 10000 nM T89213 C85LYP 11430418 IC50 > 1000 nM T89213 CQ9LX3 11560009 Ki = 50 nM T89213 CQ49SB 11640844 Ki = 30 nM T89213 CY9S3N 11654472 Ki = 53 nM T89213 CVDJ31 11669044 Ki = 62 nM T89213 CE6LT8 11670084 Ki = 55 nM T89213 C1YWG5 11732188 IC50 > 10000 nM T89213 CDHG65 11755611 IC50 = 2200 nM T89213 CA1NV0 11757487 IC50 = 5.5 nM T89213 C43LHB 11760541 IC50 > 10000 nM T89213 CJ5TE0 11798404 Ki = 93 nM T89213 C8MQT0 11799055 Ki = 1280 nM T89213 CF79NW 11799136 Ki = 2100 nM T89213 CKD08I 11800499 Ki = 140 nM T89213 CBCG71 11800628 Ki = 13 nM T89213 CUM43R 12071667 IC50 > 10000 nM T89213 CO82HM 12822578 IC50 = 8900 nM T89213 CM2YA1 15338882 Ki = 33 nM T89213 COS15P 15383694 Ki = 297 nM T89213 C7WC6U 15383696 Ki = 1750 nM T89213 CPKX57 15383697 Ki = 1135 nM T89213 CI78JL 15383698 Ki = 594 nM T89213 CJ46WB 15421872 Ki = 335 nM T89213 CF0G4N 16201612 IC50 = 4.7 nM T89213 CJV1H0 19426744 Ki = 234 nM T89213 C7U4CW 19426753 Ki = 129 nM T89213 C92QKE 19426755 Ki = 892 nM T89213 C8QZE6 19426760 Ki = 93 nM T89213 CMYK04 19426761 Ki = 119 nM T89213 CSN81D 19426762 Ki = 58 nM T89213 C3D2LV 20556258 IC50 = 60000 nM T89213 CIYU59 20587808 IC50 > 10000 nM T89213 C4Q8KN 21129772 Ki = 4.6 nM T89213 CI9M7E 21188477 Ki = 1630 nM T89213 C25DNZ 21188508 Ki = 109 nM T89213 CH06YV 21188533 Ki = 5.7 nM T89213 CKFU96 21188571 Ki = 52 nM T89213 CAGH69 21188602 Ki = 29 nM T89213 C18VHO 21188661 Ki = 21 nM T89213 CG8N0F 21188674 Ki = 88 nM T89213 C5MS6Y 21188717 Ki = 29 nM T89213 CEYW89 21188733 Ki = 57 nM T89213 CO4C3S 21336489 Ki = 17179 nM T89213 CT4PH1 21336493 Ki = 23714 nM T89213 CW92BC 21336495 Ki = 48697 nM T89213 CT7I6J 21336500 Ki = 3236 nM T89213 C8VR6Y 21336503 Ki = 14454 nM T89213 CH19JC 21336507 Ki = 12981 nM T89213 C89KZL 21336511 IC50 = 1300 nM T89213 CEOA23 22254020 IC50 > 1000 nM T89213 CBS20U 22254050 IC50 > 1000 nM T89213 CO32YX 22254068 IC50 > 1000 nM T89213 CHQT84 22254131 IC50 > 1000 nM T89213 CP7E2N 22325336 IC50 > 10000 nM T89213 C7GAN3 22617869 Ki = 2300 nM T89213 CG3VL7 25067562 IC50 > 10000 nM T89213 C7IH3J 25181112 Ki = 1 nM T89213 C7VID1 25211875 IC50 > 10000 nM T89213 CNU7P4 42630820 IC50 > 10000 nM T89213 C3MR8P 44229544 IC50 = 38000 nM T89213 CGPI02 44229545 IC50 = 15000 nM T89213 C83NXZ 44229546 IC50 = 70000 nM T89213 CQ4TG8 44229547 IC50 = 21000 nM T89213 CUVJ20 44229621 IC50 = 22000 nM T89213 CLX51J 44249749 Ki > 6309.57 nM T89213 CT4J7P 44271460 IC50 = 1000 nM T89213 CX93WE 44271463 IC50 = 8000 nM T89213 CADP10 44287730 IC50 = 21800 nM T89213 C1GH5F 44287731 IC50 = 11500 nM T89213 C40LKF 44287829 IC50 = 76000 nM T89213 CQM6N0 44287923 IC50 = 8100 nM T89213 CVJ1N7 44287924 IC50 = 7500 nM T89213 C6KR1Y 44287938 IC50 = 11900 nM T89213 CHT17W 44287971 IC50 = 900 nM T89213 C2IXS5 44287982 IC50 = 2400 nM T89213 C06XEM 44287998 IC50 = 1400 nM T89213 C7X5DG 44287999 IC50 = 150 nM T89213 C8JDU3 44288022 IC50 = 1000 nM T89213 CF79DZ 44288023 IC50 = 21000 nM T89213 CFLD69 44288053 IC50 = 3750 nM T89213 C1FW4N 44288067 IC50 = 280 nM T89213 CAI9T7 44288112 IC50 = 19 nM T89213 CJ25GY 44288137 IC50 = 2500 nM T89213 CD8G2N 44288140 IC50 = 110 nM T89213 CO4NV0 44288235 IC50 = 1100 nM T89213 C4PJG7 44288236 IC50 = 51000 nM T89213 CU2CL7 44288257 IC50 = 22300 nM T89213 CXD46O 44288311 IC50 = 12000 nM T89213 C4CT8M 44288312 IC50 > 10000 nM T89213 CEP63F 44288313 IC50 = 100 nM T89213 CN76WT 44288390 IC50 = 81 nM T89213 CS1FG8 44288395 IC50 = 3000 nM T89213 CR9V2W 44294315 IC50 = 35 nM T89213 CBKX84 44294383 IC50 = 30 nM T89213 CL4SF1 44294458 IC50 = 8.4 nM T89213 CZ8M4U 44294462 IC50 = 16 nM T89213 CHP5V6 44294463 IC50 = 237 nM T89213 C5RH2E 44294503 IC50 = 29 nM T89213 C52RAT 44294516 IC50 = 55 nM T89213 CA9O1C 44294522 IC50 = 11 nM T89213 CS9N4T 44294529 IC50 = 17 nM T89213 CX6NL7 44294536 IC50 = 1.4 nM T89213 CIG5L0 44294538 IC50 = 12 nM T89213 C9G8BI 44294543 IC50 = 63 nM T89213 CYJ67N 44294563 IC50 = 17 nM T89213 C9BNX0 44294564 IC50 = 6.5 nM T89213 CPW2U9 44294565 IC50 = 20 nM T89213 C58KAP 44294626 IC50 = 72 nM T89213 C4WNE1 44294671 IC50 = 234 nM T89213 CP1H8Y 44294672 IC50 = 33 nM T89213 CQF2Y1 44294698 IC50 = 11 nM T89213 CZV6U3 44294942 Ki = 7300 nM T89213 CY7C1N 44296638 Ki > 10000 nM T89213 CPQ8W7 44296639 Ki > 10000 nM T89213 CV75KH 44296660 Ki > 10000 nM T89213 CY8RP9 44296714 Ki > 10000 nM T89213 C4XDF3 44296729 Ki = 1250 nM T89213 CH92EK 44296730 Ki > 10000 nM T89213 CU9M0F 44296783 Ki > 10000 nM T89213 C3JU7K 44296799 Ki > 10000 nM T89213 C7Z5IK 44296819 Ki > 10000 nM T89213 C37UHB 44322256 Ki > 10000 nM T89213 CMR59C 44322264 Ki > 10000 nM T89213 CEU40C 44342355 IC50 < 1 nM T89213 C5V0ET 44342972 IC50 = 110 nM T89213 CTX16Q 44351135 Ki = 210 nM T89213 C1NUA7 44351136 Ki = 60 nM T89213 CD87HA 44351182 Ki = 410 nM T89213 CNOB51 44351197 Ki = 5.1 nM T89213 C18IMD 44362352 Ki = 11 nM T89213 C1Q0NW 44362387 Ki = 29 nM T89213 C57QXM 44362398 Ki = 3700 nM T89213 C7S1ZC 44362410 Ki = 120 nM T89213 C8IU0P 44362411 Ki = 120 nM T89213 CJ81SI 44362412 Ki = 740 nM T89213 CVJ0W5 44362444 Ki = 2420 nM T89213 COF21J 44362459 Ki = 2430 nM T89213 CPU1Q0 44362460 Ki = 660 nM T89213 CY0WE8 44362506 Ki = 172 nM T89213 C19HXB 44362526 Ki = 2190 nM T89213 CN7S5I 44362542 Ki = 260 nM T89213 CFY85W 44362553 Ki = 37 nM T89213 CPF82Y 44362574 Ki = 140 nM T89213 CRC1S0 44362610 Ki = 427 nM T89213 C14PTU 44362625 Ki = 3600 nM T89213 C9H7CY 44362626 Ki = 1260 nM T89213 C2Y4MA 44362627 Ki = 2800 nM T89213 CDW9O0 44362628 Ki = 5800 nM T89213 CC1VY8 44362637 Ki = 136 nM T89213 C49HWD 44362660 Ki = 4.5 nM T89213 CZ9LD4 44362704 Ki = 7900 nM T89213 CBWP12 44362723 Ki = 4200 nM T89213 C5HX0T 44362764 Ki = 450 nM T89213 CA53NK 44362766 Ki = 12600 nM T89213 CA39JK 44362773 Ki = 450 nM T89213 C7LEF0 44362774 Ki = 2760 nM T89213 C3J8SG 44362777 Ki = 420 nM T89213 C64OIB 44362784 Ki = 370 nM T89213 C1U7FN 44362801 Ki = 160 nM T89213 CLJ5Z4 44362810 Ki = 4000 nM T89213 CA4WM9 44362811 Ki = 2600 nM T89213 C6D4VE 44362815 Ki = 690 nM T89213 C4QJS1 44362820 Ki = 310 nM T89213 C4Y0JL 44362821 Ki = 1900 nM T89213 CM3NU2 44362822 Ki = 11100 nM T89213 CG75YO 44362830 Ki = 11 nM T89213 C1BWL6 44362831 Ki = 720 nM T89213 CY4AC7 44362832 Ki = 420 nM T89213 C9TL6E 44362838 Ki = 1700 nM T89213 CTH38K 44362839 Ki = 88000 nM T89213 C1GB9J 44362861 Ki = 380 nM T89213 COE73D 44362862 Ki = 190 nM T89213 C9MYL1 44362863 Ki = 78 nM T89213 CV58WP 44362868 Ki = 2830 nM T89213 CW7GQ3 44362878 Ki = 6500 nM T89213 CPG7J6 44362895 Ki = 3800 nM T89213 CD59JC 44362921 Ki = 12400 nM T89213 C06ZXB 44362989 Ki = 380 nM T89213 C6ZS1B 44362997 Ki = 1700 nM T89213 C2JYV1 44362998 Ki = 12000 nM T89213 CT18FD 44362999 Ki = 980 nM T89213 CLH92F 44363000 Ki = 13 nM T89213 C8ZJ1Y 44363007 Ki = 2300 nM T89213 CB26IJ 44363018 Ki = 5600 nM T89213 C4VD6X 44370176 IC50 > 10000 nM T89213 CU73FW 44370177 IC50 > 10000 nM T89213 CVN1P2 44370179 IC50 > 10000 nM T89213 C1UQR5 44370180 IC50 > 10000 nM T89213 C2D7YV 44370202 IC50 > 10000 nM T89213 CH8QJ6 44370214 IC50 > 10000 nM T89213 C7HF2B 44370215 IC50 > 10000 nM T89213 CV82UW 44370240 IC50 > 10000 nM T89213 CKGN86 44370250 IC50 > 10000 nM T89213 CF65OZ 44370266 IC50 > 10000 nM T89213 C4M5YB 44370270 IC50 > 10000 nM T89213 C4O9JP 44372383 Ki = 0.132 nM T89213 CF7B1I 44372384 Ki = 0.112 nM T89213 CUD74V 44372422 Ki = 0.183 nM T89213 CJ3UW4 44372508 Ki = 0.313 nM T89213 C1VI7M 44372691 Ki = 0.361 nM T89213 C5HBY8 44372692 Ki = 0.191 nM T89213 C4V3PB 44372750 Ki = 0.106 nM T89213 C9GPV2 44372775 Ki = 1.62 nM T89213 C45NVC 44372776 Ki = 0.285 nM T89213 CAPG42 44372777 Ki = 1.63 nM T89213 C09VWK 44372820 Ki = 1.61 nM T89213 C6H8MY 44372858 Ki = 0.393 nM T89213 C0YEK7 44373119 Ki = 0.29 nM T89213 C4IFK7 44373122 Ki = 0.707 nM T89213 C2V4JB 44373166 Ki = 0.829 nM T89213 C2YL1N 44373216 Ki = 4.5 nM T89213 CA1F2O 44377440 IC50 = 17000 nM T89213 C8D6VU 44377450 IC50 = 14000 nM T89213 CK3B4D 44377452 IC50 = 29000 nM T89213 CUEY97 44377460 IC50 = 15000 nM T89213 C87OLK 44377461 IC50 = 18000 nM T89213 C94TQS 44377468 IC50 = 8500 nM T89213 CW32ZL 44377689 IC50 = 19000 nM T89213 CO7RQ6 44377722 IC50 = 2800 nM T89213 CR0I6K 44377731 IC50 = 35000 nM T89213 C0TK1X 44377854 IC50 = 22000 nM T89213 CG40NV 44396821 IC50 = 2 nM T89213 C8TO9E 44396885 IC50 = 4 nM T89213 CNX26W 44409121 IC50 = 22.39 nM T89213 CP8UY4 44409155 IC50 = 97.72 nM T89213 CE95HU 44409158 IC50 = 100 nM T89213 CNJ4L1 44409161 IC50 = 1862.09 nM T89213 CV8U3O 44409173 IC50 = 3890.45 nM T89213 CA9D4U 44409177 IC50 = 33.88 nM T89213 CIX5R1 44409191 IC50 = 25118.86 nM T89213 CEQ1A7 44409205 IC50 = 1318.26 nM T89213 C2E9GT 44409209 IC50 = 7244.36 nM T89213 CG5V6C 44409210 IC50 = 15848.93 nM T89213 CPZ29J 44409234 IC50 = 436.52 nM T89213 CJT9I2 44409236 IC50 = 3388.44 nM T89213 CQI2G4 44409237 IC50 = 186.21 nM T89213 CU98VX 44409242 Ki = 100 nM T89213 CM9XR2 44409268 IC50 = 239.88 nM T89213 CG2HR8 44409307 IC50 = 645.65 nM T89213 CKYH61 44409330 IC50 = 331.13 nM T89213 CLO9A4 44409340 IC50 = 93.33 nM T89213 CN06IW 44409345 IC50 = 48.98 nM T89213 C8C9KV 44409363 IC50 = 776.25 nM T89213 CMDI45 44409367 IC50 = 37.15 nM T89213 CR9L3M 44439430 IC50 = 16 nM T89213 CG9YZ6 44439431 IC50 = 11 nM T89213 C9R2MW 44439432 IC50 = 51 nM T89213 CLS72Z 44439433 IC50 = 28 nM T89213 C35DFS 44439434 IC50 = 53 nM T89213 CF53VL 44439435 IC50 = 95 nM T89213 C9XJ6T 44439436 IC50 = 107 nM T89213 CRM71L 44439437 IC50 = 186 nM T89213 CDT59H 44439438 IC50 = 43 nM T89213 C54LYI 44439439 IC50 = 14 nM T89213 C38VQO 44439440 IC50 = 50 nM T89213 CBY8K1 44439441 IC50 = 832 nM T89213 CXHI64 44439442 IC50 = 9772 nM T89213 CVM17U 44439443 IC50 = 2882 nM T89213 C6SRX4 44439444 IC50 = 1905 nM T89213 C1K6RQ 44439445 IC50 = 7762 nM T89213 C1HAV7 44439446 IC50 = 871 nM T89213 CGU62P 44439456 IC50 = 467 nM T89213 CLC65I 44439485 IC50 = 50 nM T89213 C27RMO 44439486 IC50 = 191 nM T89213 CL72NO 44439489 IC50 = 263 nM T89213 CH4ME0 44439491 IC50 = 1862 nM T89213 CT5WQ2 44439493 IC50 = 12022 nM T89213 CJM96N 44461116 IC50 > 30000 nM T89213 C4DL5C 44469677 IC50 > 10000 nM T89213 C68NXC 44517723 Ki = 22 nM T89213 C90GPQ 44563341 Ki = 12 nM T89213 CG0VZ9 44563342 Ki = 27 nM T89213 CZ65XF 44579887 IC50 > 10000 nM T89213 CVO10S 44580050 IC50 > 10000 nM T89213 CF4PM0 45267382 IC50 = 13000 nM T89213 C51LCW 45267391 IC50 > 1000000 nM T89213 CFY4R2 45267593 Ki = 160 nM T89213 CTB32R 45268225 IC50 = 16000 nM T89213 C4DZO1 45268459 Ki = 42 nM T89213 CQ7J4A 45268477 Ki = 210 nM T89213 C9IJK8 45268483 Ki = 43 nM T89213 CC8P5K 45269117 IC50 = 9000 nM T89213 C6ETI8 45269118 IC50 = 15000 nM T89213 CX53RU 45269119 IC50 = 320000 nM T89213 CRN8Y1 45269121 IC50 = 4300 nM T89213 CED18G 45269300 Ki = 330 nM T89213 CZC09M 45269305 Ki = 49 nM T89213 CFJ17A 45269306 Ki = 18 nM T89213 CCQ8W4 45269310 Ki = 3000 nM T89213 CNA70T 45269316 Ki = 7.3 nM T89213 C1SB8A 45269317 Ki = 15 nM T89213 CDM73H 45270136 Ki = 32 nM T89213 C2Q4SM 45270142 Ki = 120 nM T89213 CLPB92 45270153 Ki = 150 nM T89213 CGXC75 45270156 Ki = 790 nM T89213 C0R5NB 45270796 IC50 = 21000 nM T89213 CZ9OC8 45270973 Ki = 7.4 nM T89213 CB94YA 45270992 Ki = 1100 nM T89213 CBW87K 45271004 Ki = 27 nM T89213 C08OEP 45271626 IC50 = 32000 nM T89213 CE8Z1K 45271821 Ki = 24 nM T89213 C1L4DN 45271828 Ki = 890 nM T89213 CLD3T9 45271838 Ki = 45 nM T89213 CP7K0V 45271861 Ki = 44 nM T89213 C5R7OL 45272520 IC50 = 25000 nM T89213 C5DE4U 45272692 Ki = 29 nM T89213 C1JLQ3 45273630 Ki = 48 nM T89213 C27VWT 45273649 Ki = 470 nM T89213 C7HQ9B 45273656 Ki = 10 nM T89213 CN84EP 45487432 IC50 = 4.3 nM T89213 C0KS4E 45487433 IC50 = 10 nM T89213 C0AJ6Z 45487434 IC50 = 0.46 nM T89213 CM3WY0 45487435 IC50 = 0.27 nM T89213 C6LP8J 45487440 IC50 = 0.56 nM T89213 C6QZC0 45487445 IC50 = 1.8 nM T89213 C2DEU0 45487446 IC50 = 19 nM T89213 C30LDO 45487447 IC50 = 0.2 nM T89213 CL9PW1 45487448 IC50 = 0.13 nM T89213 CLW68C 45487464 IC50 = 0.69 nM T89213 CKZ8G4 45487489 IC50 = 0.27 nM T89213 CDI5O1 45487490 IC50 = 0.16 nM T89213 CDN4B9 45487501 IC50 = 8 nM T89213 CUQ3E0 45487511 IC50 = 21 nM T89213 CF51BR 45487512 IC50 = 7.7 nM T89213 C6P8XL 45487514 IC50 = 5.2 nM T89213 C2E3BH 45487522 IC50 = 1.5 nM T89213 CI7TE1 45487523 IC50 = 1.7 nM T89213 CA34QJ 45487524 IC50 = 0.39 nM T89213 C1JK8M 46231121 Ki = 63 nM T89213 CZ6UR9 46231123 Ki = 275 nM T89213 C5YB1P 46231125 Ki = 5 nM T89213 CPU4M0 46231127 Ki = 128 nM T89213 CE53PU 46231128 Ki = 7 nM T89213 CXB60L 46879453 Ki = 3460 nM T89213 C6I9DP 46879454 Ki = 3990 nM T89213 CW2A3H 46879455 Ki = 1060 nM T89213 CQXC46 46879456 Ki = 1670 nM T89213 CZL0Q8 46879457 Ki = 1120 nM T89213 C8B7EU 46879521 Ki = 1240 nM T89213 C2UNT0 46879522 Ki = 5250 nM T89213 CH64ZP 46879523 Ki = 5920 nM T89213 CI02OK 46879524 Ki = 3640 nM T89213 C3J4IO 46879560 Ki = 221 nM T89213 CI8PV4 46879563 Ki = 616 nM T89213 C2U6ET 46879606 Ki = 1250 nM T89213 CGYM19 46879607 Ki = 318 nM T89213 COC16Y 46879608 Ki = 342 nM T89213 CMQ71F 46879609 Ki = 3300 nM T89213 C9KUH0 46879610 Ki = 5200 nM T89213 CNU02D 46879646 Ki = 316 nM T89213 C7MNC2 46879649 Ki = 379 nM T89213 C93GXU 46879650 Ki = 153 nM T89213 COCW38 46879690 Ki = 482 nM T89213 CV3H9P 46879691 Ki = 69 nM T89213 CLS02W 46879692 Ki = 712 nM T89213 CEC8Y3 46879693 Ki = 175 nM T89213 CBV32D 46879737 Ki = 2550 nM T89213 CEJ2S6 46879779 Ki = 195 nM T89213 CW76YJ 46879780 Ki = 332 nM T89213 CMC83J 46879781 Ki = 55 nM T89213 CQS25A 46879822 Ki = 122 nM T89213 C09QEC 46879823 Ki = 107 nM T89213 C1QOS3 46879824 Ki = 956 nM T89213 C0EQ5P 46879876 Ki = 464 nM T89213 CZD7T5 46880224 Ki = 248 nM T89213 CTZP80 46934142 Ki = 0.9 nM T89213 C7AT5K 49797585 Ki = 6.1 nM T89213 C9VLN4 49797586 Ki = 49 nM T89213 CE2J0G 49865799 Ki = 1500 nM T89213 C9EKQ2 49865800 Ki = 460 nM T89213 C56RHM 49865801 Ki = 270 nM T89213 CDXJ84 49865803 Ki = 59 nM T89213 CK4P7T 49865804 Ki = 40 nM T89213 C3K6UN 49865805 Ki = 110 nM T89213 CC5A6O 49865807 Ki = 260 nM T89213 C1MHQ2 49865808 Ki = 3 nM T89213 C3AV6E 49865809 Ki = 6.7 nM T89213 CEHU78 49865810 Ki = 41 nM T89213 CJ14FC 49865811 Ki = 73 nM T89213 CY7E6O 49865812 Ki = 130 nM T89213 C9DJ0C 49865813 Ki = 51 nM T89213 CGO62F 50925473 Ki > 6309.57 nM T89213 CH5A3Z 52953217 Ki = 22 nM T89213 CV10HR 52953219 Ki = 26 nM T89213 CHT4P6 53359565 Ki = 400 nM T89213 CXH0Z7 54580352 Ki = 42 nM T89213 CB98NS 54580549 Ki = 38 nM T89213 C1MQ6W 54581330 Ki = 50 nM T89213 CIKW16 54582342 Ki = 29 nM T89213 C97QRD 54582344 Ki = 4.3 nM T89213 C47JQY 54582347 Ki = 150 nM T89213 CO9CV6 54582349 Ki = 96 nM T89213 CN4PI1 54583329 Ki = 13 nM T89213 CG4XK9 54583331 Ki = 130 nM T89213 CA4YQ3 54583518 Ki = 5 nM T89213 CRB0H2 54583519 Ki = 141 nM T89213 C7MAQ6 54584288 Ki = 38 nM T89213 C5QT0M 54584289 Ki = 24 nM T89213 C19USF 54585270 Ki = 130 nM T89213 CQOS61 54586207 Ki = 97 nM T89213 CJF4D5 54587217 Ki = 19 nM T89213 CUY61J 54587218 Ki = 23 nM T89213 C7O6CY 54587220 Ki = 38 nM T89213 CVRU23 54587222 Ki = 140 nM T89213 C6OPM3 54587431 Ki = 22 nM T89213 CLQ9Y2 56841989 EC50 = 0.1 nM T89213 CSGN50 57384007 IC50 = 62 nM T89213 CN9L4K 57404430 Ki > 10000 nM T89213 C74WIF 62706260 IC50 = 2200 nM T89213 CVP39A 62706261 IC50 = 1300 nM T89213 CE08IH 62706262 IC50 = 300 nM T89213 C4Y6CQ 62706421 IC50 = 190 nM T89213 C1WO2F 62706422 IC50 > 10000 nM T89213 C7NXW4 62706423 IC50 = 460 nM T89213 C7TSV1 62706424 IC50 = 170 nM T89213 CR2T9J 62706425 IC50 = 550 nM T89213 C0C6HL 62706426 IC50 = 180 nM T89213 C0B5HQ 70686176 Ki = 15 nM T89213 C1YB4T 71456264 IC50 = 4.7 nM T89213 CGKU71 71717895 Ki = 42 nM T89213 C8QO1W 71719108 Ki > 5000 nM T89213 CGHY58 71719788 IC50 = 9.8 nM T89213 C9UH7J 72205287 Ki = 7.3 nM T89213 CD18YC 72205289 Ki = 31 nM T89213 C70RKE 72205291 Ki = 9.9 nM T89213 CL8NG4 72205482 Ki = 200 nM T89213 CDZU03 72205484 Ki > 5000 nM T89213 CH2VP3 72205486 Ki = 130 nM T89213 CAK56G 72205667 Ki = 41 nM T89213 C3NVQ7 72205669 Ki = 890 nM T89213 CBL6T0 72205671 Ki = 14 nM T89213 C4W1IA 72205853 Ki = 73 nM T89213 CA26US 72205877 Ki > 5000 nM T89213 CFC0Q6 72206048 Ki > 5000 nM T89213 CWH6T3 72548703 IC50 = 0.13 nM T89213 CFV1X0 72711815 Ki > 1000 nM T89213 CE6KV1 72712030 Ki > 1000 nM T89213 C7V2BT 72714999 IC50 = 42 nM T89213 CL53DX 72715000 IC50 = 54 nM T89213 CFQY96 73345485 Ki > 1000 nM T89213 CRU6C1 73345939 IC50 > 10000 nM T89213 CK9QD3 73345940 IC50 > 10000 nM T89213 C1X2AR 73346549 Ki > 5000 nM T89213 CJ5HR8 73347019 Ki = 220 nM T89213 C2TWI4 73348990 IC50 = 5032 nM T89213 CYID03 73348991 IC50 > 10000 nM T89213 C3Y8HL 73349568 Ki = 86 nM T89213 CPXJ28 73349570 Ki > 5000 nM T89213 C1NQ7B 73350103 Ki > 1000 nM T89213 CTJ3D0 73350105 Ki = 230 nM T89213 CU94RO 73350550 IC50 = 4380 nM T89213 C7CMG0 73350551 IC50 > 10000 nM T89213 C8TJU9 73350552 IC50 > 10000 nM T89213 C0NM1P 73351119 Ki > 1000 nM T89213 CM5ZV2 73351127 Ki = 1000 nM T89213 C7TL4C 73352596 Ki = 77 nM T89213 C27BRN 73352597 Ki = 63 nM T89213 CB9R8P 73353058 Ki = 130 nM T89213 CO4GL8 73353059 Ki > 1000 nM T89213 C2Z1JL 73353529 IC50 = 265 nM T89213 C18MUR 73353531 IC50 = 4270 nM T89213 C28UNZ 73353532 IC50 = 892 nM T89213 C10OEC 73353533 IC50 = 62 nM T89213 CRC73X 73354075 Ki > 1000 nM T89213 CRL10F 73354088 Ki > 5000 nM T89213 CL5A3F 73354090 Ki = 360 nM T89213 CIFL82 73354092 Ki > 5000 nM T89213 C9XCU8 73354094 Ki > 5000 nM T89213 C34SQD 73354098 Ki > 5000 nM T89213 CCK72G 73355613 Ki > 5000 nM T89213 C4FDT1 73355615 Ki = 71 nM T89213 CO26NJ 73355617 Ki = 30 nM T89213 C1WH4P 73356587 IC50 > 10000 nM T89213 CUM6D5 73357147 Ki > 1000 nM T89213 CXJ85A 73357158 Ki = 1200 nM T89213 CB3FG4 85472343 Ki = 930 nM T89213 CK5B7R 118718116 Ki = 0.9 nM T89213 C94LWU 118718124 Ki = 14 nM T89213 CJ5Q9R 118718125 Ki = 4.5 nM T89213 C92ZVT 118718320 Ki = 260 nM T89213 CW2BG8 127029975 Ki = 720 nM T89213 C7Q2WP 127030359 Ki = 360 nM T89213 CK0A1M 127031281 Ki = 410 nM T89213 C0XR6M 127041306 IC50 = 0.1047 nM T89213 C7GL1W 127041307 Ki = 4.5 nM T89213 CIQ8P1 127041308 Ki = 4 nM T89213 C52YJP 127041902 Ki = 6.9 nM T89213 C24LXZ 127041903 Ki = 3.1 nM T89213 CH64EZ 127041904 Ki = 41 nM T89213 C5PA2G 127041908 Ki = 0.34 nM T89213 C7TM1Y 127042243 Ki = 22 nM T89213 C62JIE 127042244 Ki = 0.077 nM T89213 CWP0V5 136216703 Ki = 4200 nM T89213 CL53MA 145948574 Ki = 0.41 nM T89213 CP0FM6 145948575 Ki > 1000 nM T89213 CG8SN7 145965939 EC50 > 1000 nM T89213 C8ZAN2 145979152 EC50 = 15.85 nM T89213 C4SB9P 145979291 EC50 > 1000 nM T89213 CQ78WY 145979469 Ki = 10000 nM T89213 CO1M3D 145979616 Ki = 3981.07 nM T89213 C3OXL9 145979975 Ki = 5000 nM T89213 C4H9BZ 145980763 Ki = 398.11 nM T89213 CH5MZ8 145980782 EC50 = 316.23 nM T89213 CI5F7E 145980802 Ki > 10000 nM T89213 CP4RI5 145980997 EC50 = 0.1995 nM T89213 CW80EN 145981168 Ki > 10000 nM T89213 CTF1C6 145981319 Ki = 1995.26 nM T89213 COB75I 145981742 Ki = 500 nM T89213 C60AUT 145981829 EC50 > 1000 nM T89213 COF9U8 145982156 Ki > 10000 nM T89213 CXE2K1 145984150 EC50 = 316.23 nM T89213 CM4VG2 145984378 EC50 = 79 nM T89213 CG74XB 145985156 Ki = 1000 nM T89213 C5XL9U 145985176 EC50 > 30 nM T89213 C63DRI 145985639 Ki > 10000 nM T89213 C5UDH2 145986414 Ki = 2500 nM T89213 CLEQ40 145986472 EC50 = 15.85 nM T89213 CZ68SU 145986539 Ki > 10000 nM T89213 CGB4Y3 145987289 Ki > 10000 nM T89213 CI1XY0 145987577 Ki = 5000 nM T89213 C4T5IJ 145987618 Ki > 10000 nM T89213 CL2I3Y 145987802 Ki = 10000 nM T89213 CIZ94Y 145988210 Ki = 3.981 nM T89213 CRW15D 145989250 Ki = 1258.93 nM T89213 C5O8AZ 145989327 EC50 > 1000 nM T89213 CG63IW 145989789 Ki = 6300 nM T89213 CF5OV2 145990257 EC50 > 1000 nM T89213 CH50MF 145991293 EC50 > 1000 nM T89213 CDX86E 145991438 Ki = 1584.89 nM T89213 C6PS8F 145991876 EC50 > 1000 nM T89213 C7K8CT 145992181 EC50 = 0.1995 nM T89213 CC72HP 145992661 EC50 = 0.1995 nM T89213 C5KF0O 145992989 Ki = 199.53 nM T89213 CQH29C 145993358 Ki = 12.59 nM T89213 C9Z4PM 145993376 Ki > 10000 nM T89213 CAZ6I7 145993698 EC50 = 125.89 nM T89213 CPD7M9 145994220 EC50 > 1000 nM T89213 C4AB9K 155512045 IC50 = 234.42 nM T89213 CHW62U 155517347 IC50 = 489.78 nM T89213 C4KN0H 155517812 Ki = 0.3631 nM T89213 C2BUO8 155523949 Ki = 0.257 nM T89213 CQF01J 155524657 IC50 = 363.08 nM T89213 CY8MK6 155533017 Ki = 25.12 nM T89213 C2VJ4Y 155537755 Ki = 0.2754 nM T89213 C2GBO9 155541756 Ki = 0.5754 nM T89213 CCK32B 155543070 Ki = 400 nM T89213 C5A7BF 155546907 Ki = 8.128 nM T89213 CCZ09U 155547323 Ki = 1600 nM T89213 C1T7DH 155549336 Ki = 290 nM T89213 CDT81L 155553742 Ki > 3000 nM T89213 CX43VE 155561277 Ki > 10000 nM T89213 C4M9NL 155561620 Ki = 1400 nM T89213 C86FRY 155563387 Ki = 2.344 nM T89213 CH4XA1 155564444 Ki = 31.62 nM T89213 CC8WB6 155565033 Ki = 12.88 nM T89213 D00OLA 44409453 Ki = 30 nM T89213 D05ZUX 44207909 Ki >= 1000 nM T89213 D07OOG 73347134 Ki = 80 nM T89213 D07XFL 10007341 IC50 = 9600 nM T89213 D08YWE 73348635 Ki = 120 nM T89213 D0G4HT 73354703 Ki = 7.5 nM T89213 D0J9VA 44409452 Ki = 220 nM T89213 D0N6HL 10052173 IC50 = 12000 nM T89213 D0Q2IU 44439563 Ki > 1000 nM T89213 D0T2RY 9948320 Ki >= 1000 nM T89213 D0U5TK 5311022 Ki = 0.25 nM T89213 D0V0HM 73345612 Ki = 140 nM T82393 D00MDP 466151 IC50 = 5.5 nM T82393 D05VZE 119031 Ki = 0.4 nM T82393 D0HG5M 11452716 IC50 = 125.89 nM T82393 D0MW3H 9824350 Ki = 230 nM T82393 D03ESO 216470 IC50 = 40 nM T82393 D01DVX 9847838 IC50 = 0.2 nM T82393 D03BOZ 3342298 IC50 = 14 nM T82393 D05VNG 9908389 IC50 = 0.2 nM T82393 D0E5GY 9904965 IC50 = 20 nM T82393 D0H5CD 5748217 IC50 = 1.8 nM T82393 D0P8YC 5362422 IC50 = 0.4 nM T82393 D0T9HG 132519 IC50 = 7.5 nM T82393 C4D7TS 448002 IC50 = 2300 nM T82393 CC5O4E 4369384 IC50 = 4300 nM T82393 CW5SE3 5288615 IC50 = 8 nM T82393 C5OMB7 6102708 IC50 = 67 nM T82393 C0M3LR 6323382 IC50 = 8 nM T82393 CA0ZH1 9798114 IC50 = 10 nM T82393 C78EKW 9798637 IC50 = 23 nM T82393 C76RCQ 9801569 IC50 = 2 nM T82393 CM9GH8 9802180 IC50 = 103 nM T82393 CJY12B 9802219 IC50 = 4800 nM T82393 C4CN0H 9802436 Ki = 6.2 nM T82393 C40THQ 9802812 IC50 = 42000 nM T82393 C83FVW 9803207 IC50 = 413 nM T82393 C3QS5H 9803407 IC50 = 90 nM T82393 C4QCG9 9803771 IC50 = 6 nM T82393 C23VTC 9804342 IC50 = 6 nM T82393 C49HNU 9805016 IC50 = 272 nM T82393 CP65QD 9805079 IC50 = 2650 nM T82393 CXSU10 9805304 IC50 = 7 nM T82393 CO4D0U 9805473 IC50 = 13 nM T82393 CT8X1F 9806970 IC50 = 66 nM T82393 C76CKA 9807105 IC50 = 840 nM T82393 C67XKV 9808391 IC50 = 138 nM T82393 CS07BM 9808594 IC50 = 124 nM T82393 C1VT4J 9819974 IC50 = 5 nM T82393 CQG86S 9820708 IC50 = 594 nM T82393 CTF8V4 9823391 IC50 > 3000 nM T82393 CY1H0O 9824331 IC50 = 14 nM T82393 CUZ25T 9825237 IC50 = 17 nM T82393 CXL65P 9825920 IC50 = 403 nM T82393 CVSJ72 9826275 IC50 = 208 nM T82393 C7W3TG 9826481 IC50 = 12 nM T82393 CPW60S 9827023 IC50 = 20 nM T82393 CZ7D6M 9827273 IC50 = 8100 nM T82393 C3SZ8Y 9827469 IC50 = 4950 nM T82393 C24CZI 9827635 IC50 = 33 nM T82393 C2TU0C 9827807 IC50 = 271 nM T82393 CL59JS 9827846 IC50 = 4.3 nM T82393 C7I2FO 9828039 IC50 = 420 nM T82393 C8WH1Q 9840355 IC50 = 626 nM T82393 CEAZ87 9840395 IC50 = 38 nM T82393 CQ5L0D 9842167 IC50 = 75 nM T82393 CH63ZI 9842332 IC50 = 3 nM T82393 CEB90C 9846418 IC50 = 154 nM T82393 CWY1J9 9846501 IC50 = 1500 nM T82393 CI7T1S 9846676 IC50 = 2.5 nM T82393 C0KP9H 9847092 IC50 = 565 nM T82393 CA1IP0 9847191 IC50 > 3000 nM T82393 C20UBL 9847528 IC50 = 1300 nM T82393 CG14CO 9848625 IC50 = 47 nM T82393 CX3EW2 9849576 IC50 = 65 nM T82393 CHVL24 9849957 IC50 = 386 nM T82393 C9P1BH 9851086 IC50 = 581 nM T82393 CC70WV 9858468 IC50 = 17 nM T82393 CR37HQ 9861014 IC50 = 120 nM T82393 CXZ1R9 9861547 Ki = 33 nM T82393 CU51IV 9865936 IC50 = 229 nM T82393 CR10NL 9866770 IC50 = 8700 nM T82393 C0E7JQ 9866988 IC50 = 188 nM T82393 C6EZ1V 9867022 IC50 = 14 nM T82393 CP4Y7O 9867411 IC50 = 7 nM T82393 C2L9SU 9868329 IC50 = 95 nM T82393 CJS23I 9868333 IC50 = 150 nM T82393 C5O0GC 9868490 IC50 = 28 nM T82393 CRI23M 9868515 IC50 = 11 nM T82393 C4K2GH 9868577 IC50 = 170 nM T82393 C4ZR7O 9868713 IC50 = 16 nM T82393 CT76IN 9869441 IC50 = 115 nM T82393 CA6G0W 9869598 IC50 = 270 nM T82393 CZO6K4 9869819 IC50 = 95 nM T82393 C5ELS6 9869902 IC50 = 72 nM T82393 C25-SEP 9870933 IC50 = 34 nM T82393 C4JQ7A 9871823 IC50 = 188 nM T82393 CU9L3X 9879183 IC50 = 157 nM T82393 C0ZT7A 9883002 Ki = 3700 nM T82393 C4PB5Z 9887544 IC50 = 1200 nM T82393 CFG4Q2 9887831 IC50 = 9 nM T82393 CC87LP 9888280 IC50 = 222 nM T82393 C8AJB7 9888429 IC50 = 2400 nM T82393 CD76WB 9888485 IC50 = 250 nM T82393 CB2YG7 9889128 IC50 = 197 nM T82393 CNX78A 9890733 IC50 = 301 nM T82393 CMD0S2 9891009 IC50 = 294 nM T82393 CN0MS4 9891048 IC50 = 5 nM T82393 CR50BS 9892336 IC50 = 82 nM T82393 C1KV7J 9892518 IC50 = 207 nM T82393 CK1F3O 9892889 IC50 = 6830 nM T82393 C2G5AQ 9894201 IC50 = 29 nM T82393 CH8O4Q 9894447 IC50 = 393 nM T82393 C97GSC 9903557 Ki > 1000 nM T82393 CMSC52 9908418 IC50 > 10000 nM T82393 CKWF30 9908681 IC50 = 13 nM T82393 CVT4D1 9910032 IC50 = 20 nM T82393 CPO8V1 9910282 IC50 = 6.31 nM T82393 C4E6LR 9910544 IC50 = 6 nM T82393 CT50EC 9912183 IC50 = 1560 nM T82393 C2GMQ0 9912235 IC50 = 12 nM T82393 CRNL01 9912879 IC50 = 55 nM T82393 C8VJ9Z 9913053 IC50 = 277 nM T82393 CI5A3G 9913301 IC50 = 273 nM T82393 CX1Q5C 9913489 IC50 = 631 nM T82393 C8AQ3S 9913990 IC50 = 1 nM T82393 CU9B3E 9914147 IC50 = 43 nM T82393 CX3C2G 9914326 IC50 = 149 nM T82393 CM39FU 9915194 IC50 = 346 nM T82393 CM7UO8 9924798 IC50 = 180 nM T82393 CBPD13 9926779 IC50 = 145 nM T82393 CSA12Z 9927353 IC50 = 73 nM T82393 C02JVU 9928154 IC50 = 1.5 nM T82393 C7EIX4 9930068 IC50 = 6500 nM T82393 CLJ61Q 9931505 IC50 = 880 nM T82393 CJI5A7 9932167 IC50 = 270 nM T82393 C1I2FW 9932632 IC50 = 1100 nM T82393 C3VO2E 9932958 IC50 = 40000 nM T82393 CT2KM9 9933083 IC50 = 30 nM T82393 C2EUL8 9933259 IC50 = 14 nM T82393 CF26MY 9934052 IC50 > 10000 nM T82393 CA5V8M 9934053 IC50 > 3000 nM T82393 CGJZ78 9934997 IC50 = 10 nM T82393 CDRC76 9936405 IC50 = 808 nM T82393 CH9G5D 9936469 IC50 = 59 nM T82393 C68MQN 9936625 IC50 = 9100 nM T82393 C7GJF8 9936712 IC50 = 26 nM T82393 CG38KL 9936728 IC50 = 67 nM T82393 CX7VQ9 9937188 IC50 = 96 nM T82393 CB2WS9 9944588 IC50 = 4 nM T82393 C12ZGS 9945200 IC50 = 13 nM T82393 C0MLZ6 9945553 IC50 = 105 nM T82393 C6TH4I 9947270 IC50 = 26 nM T82393 CSN61C 9948296 Ki > 1000 nM T82393 C16HTN 9948666 IC50 = 7 nM T82393 C52IUJ 9949603 IC50 = 105 nM T82393 CF1DO9 9950475 IC50 > 10000 nM T82393 COVR98 9951986 IC50 = 1 nM T82393 CQY54S 9952396 IC50 = 10000 nM T82393 C9OY4Z 9953817 IC50 = 470 nM T82393 C16GIN 9953861 IC50 = 1570 nM T82393 CR6EX3 9953909 IC50 = 1700 nM T82393 CABI45 9954117 IC50 = 43 nM T82393 C6GA8D 9954513 IC50 = 503 nM T82393 CH9YL3 9954604 IC50 = 293 nM T82393 C37VXK 9954605 IC50 = 213 nM T82393 C9X0YR 9954867 IC50 = 430 nM T82393 CMV37W 9955127 IC50 = 28 nM T82393 CQW79G 9955564 IC50 = 3 nM T82393 CWE6N8 9955640 IC50 = 104 nM T82393 C3P0EM 9955696 IC50 = 16 nM T82393 C3ZLA1 9956465 IC50 = 82 nM T82393 C56GFP 9956833 IC50 = 610 nM T82393 CQ80MP 9957107 IC50 = 318 nM T82393 C5I0VJ 9957500 IC50 = 11 nM T82393 CN76XI 9957653 IC50 = 301 nM T82393 CPJR82 9957875 IC50 = 98 nM T82393 CWE4D3 9958604 IC50 = 421 nM T82393 CNHT34 9959421 IC50 = 199 nM T82393 CV40RB 9960075 Ki = 5 nM T82393 CC4I0U 9960450 IC50 = 882 nM T82393 C9DRB7 9966028 IC50 = 17 nM T82393 CYK75X 9967932 IC50 = 28 nM T82393 C71YGT 10025307 Ki > 1000 nM T82393 C1X0SA 10041385 Ki = 274 nM T82393 CNA3G4 10042214 IC50 = 966 nM T82393 CHF92V 10047100 Ki > 1000 nM T82393 CCF5Z4 10047585 IC50 = 0.3 nM T82393 C1N9UX 10050222 IC50 = 16 nM T82393 C42YWK 10055393 IC50 = 79.43 nM T82393 CSW7B3 10067146 Ki > 1000 nM T82393 CPS4R9 10076090 IC50 = 122 nM T82393 CUT28D 10088847 Ki = 5.06 nM T82393 C7R0NY 10096444 IC50 = 16000 nM T82393 C9T2AW 10116042 IC50 = 147 nM T82393 CP5L0W 10117663 IC50 = 208 nM T82393 CU3ZM2 10118633 IC50 > 1000 nM T82393 C2F8KW 10119294 IC50 = 190 nM T82393 CPA4R9 10119730 IC50 > 1000 nM T82393 C0Q9DW 10120586 IC50 = 435 nM T82393 C0KHW5 10120930 IC50 = 124 nM T82393 CP65KL 10125869 Ki = 66 nM T82393 C0O9QV 10126803 Ki = 60 nM T82393 CY2N3D 10127629 IC50 = 855 nM T82393 C1N4MJ 10127670 IC50 = 535 nM T82393 CIL09Z 10127889 IC50 = 91 nM T82393 C07KFI 10128313 IC50 = 96 nM T82393 CB3I6K 10128659 IC50 = 160 nM T82393 C6ZK3A 10128916 IC50 = 160 nM T82393 CS54CQ 10133565 IC50 = 51 nM T82393 C0SVY1 10134897 IC50 = 201 nM T82393 CFXC89 10139040 IC50 = 37 nM T82393 CU6Y9T 10140438 IC50 = 26 nM T82393 CE75BY 10140776 IC50 = 867 nM T82393 C5DA1U 10141270 IC50 = 314 nM T82393 C5H1ZM 10141426 IC50 = 226 nM T82393 C6MSI0 10141443 IC50 = 45 nM T82393 CLXF15 10141613 IC50 > 3000 nM T82393 C7VF1K 10141614 IC50 = 102 nM T82393 CPXB21 10143028 IC50 = 54 nM T82393 CEG7Q1 10143029 IC50 > 3000 nM T82393 C9KXN5 10143180 IC50 = 240 nM T82393 C23WZR 10143587 IC50 = 2503 nM T82393 CAM6U7 10143672 IC50 > 1000 nM T82393 C82SMW 10144091 IC50 = 336 nM T82393 C9MJD2 10150046 Ki = 900 nM T82393 CD3U8E 10150649 Ki = 8 nM T82393 CZW98O 10156375 IC50 > 1000 nM T82393 CPY87U 10158366 IC50 = 119 nM T82393 CYO8D2 10159633 IC50 = 8.3 nM T82393 CQ41YI 10161391 IC50 = 480 nM T82393 CCU9S1 10162155 IC50 > 100 nM T82393 C7SXD4 10162245 IC50 = 76 nM T82393 CCM0Y8 10165180 IC50 = 161 nM T82393 CE10MK 10165419 IC50 > 1000 nM T82393 CP02FJ 10165420 IC50 > 1000 nM T82393 CWT46A 10165477 IC50 > 3000 nM T82393 C0K7HT 10165868 IC50 = 124 nM T82393 CNTC03 10172417 Ki = 12 nM T82393 C6IW4O 10173876 IC50 = 1100 nM T82393 C4QY3V 10175210 IC50 = 110 nM T82393 C5JM1A 10179045 IC50 = 39 nM T82393 CS6X2R 10183408 IC50 = 296 nM T82393 C6OE9H 10183692 IC50 = 233 nM T82393 CDM94B 10183693 IC50 = 913 nM T82393 C2GV5Q 10183755 IC50 = 17 nM T82393 CH04IS 10184457 IC50 = 160 nM T82393 C3E9NF 10184537 IC50 = 109 nM T82393 CTDP62 10184579 IC50 = 258 nM T82393 CXQ8N0 10185100 IC50 = 90 nM T82393 C2OM9G 10186288 IC50 = 401 nM T82393 CV7YI1 10186544 IC50 = 506 nM T82393 CA9FG4 10187181 IC50 = 120 nM T82393 CQY98L 10194369 Ki = 50 nM T82393 CY36NO 10196425 IC50 = 5400 nM T82393 C5CUM9 10202769 IC50 = 5.9 nM T82393 CX8BS3 10203685 IC50 = 900 nM T82393 C32RAQ 10204620 IC50 = 595 nM T82393 C7AU0H 10205886 IC50 = 627 nM T82393 CS1CA5 10207780 IC50 = 77 nM T82393 CV4DG9 10209314 IC50 = 161 nM T82393 CD76KE 10209382 IC50 = 370 nM T82393 C6M2TB 10215513 Ki = 290 nM T82393 C1C7AH 10223757 IC50 = 29 nM T82393 CLH71C 10225319 IC50 = 3.7 nM T82393 CN8MS2 10225737 IC50 > 3000 nM T82393 C2X1KF 10226116 IC50 = 223 nM T82393 CJ46HR 10227522 IC50 = 54 nM T82393 CUE63Q 10227853 IC50 = 123 nM T82393 CSDG58 10228529 IC50 = 58 nM T82393 CLJ3Y9 10230286 IC50 = 1000 nM T82393 C1ZX6C 10230907 IC50 > 3000 nM T82393 CA5F2L 10236529 Ki = 1600 nM T82393 CV9TB8 10237300 Ki = 50 nM T82393 CCTY95 10237492 IC50 = 1 nM T82393 CRF32B 10237550 Ki = 8 nM T82393 CCQ9V5 10239716 IC50 = 195 nM T82393 CL67DT 10252311 Ki = 177 nM T82393 CJKD83 10268288 IC50 = 50 nM T82393 CMNA19 10270268 IC50 = 299 nM T82393 C0K2ES 10273642 IC50 = 75 nM T82393 CES6A5 10276821 IC50 = 420 nM T82393 C0GU6B 10277568 IC50 = 298 nM T82393 CY6K1G 10277706 IC50 > 3000 nM T82393 C9OAE1 10277812 IC50 = 535 nM T82393 C6DT3Z 10278105 IC50 > 3000 nM T82393 C2UAM8 10278729 IC50 = 356 nM T82393 C6KR5M 10278934 IC50 = 589 nM T82393 C7TWG0 10289551 IC50 = 275 nM T82393 CJ63ER 10289607 IC50 = 81 nM T82393 CP0I5Y 10291146 IC50 = 74 nM T82393 CLP72J 10293348 IC50 = 113 nM T82393 CN14MI 10298369 IC50 = 109 nM T82393 C25EKM 10299665 IC50 = 632 nM T82393 C1BR6A 10300063 IC50 = 23 nM T82393 C80VEU 10300077 IC50 = 96 nM T82393 CFAU84 10301584 IC50 = 152 nM T82393 CP5AU1 10302088 IC50 = 102 nM T82393 C4R9ZK 10311997 IC50 = 84 nM T82393 CE6MB0 10312141 IC50 = 2800 nM T82393 C2U6MY 10318916 Ki = 40 nM T82393 CJ6XM1 10321516 IC50 = 124 nM T82393 CSFZ76 10325592 Ki = 13 nM T82393 CBTO07 10370226 IC50 = 212 nM T82393 CL97HT 10388523 Ki = 0.57 nM T82393 CY2G0R 10391428 IC50 = 39 nM T82393 C8Y7EZ 10393391 IC50 = 36 nM T82393 C1SJ4K 10435554 IC50 = 12 nM T82393 C7XE1L 10437629 IC50 = 12 nM T82393 CWV9Q2 10477531 IC50 = 510 nM T82393 CHG02V 10478612 IC50 = 730 nM T82393 C8C7NZ 10504593 IC50 = 0.6 nM T82393 CYQR28 10504595 IC50 = 1 nM T82393 C26NWM 10505010 IC50 = 1.2 nM T82393 CR24VM 10528406 IC50 = 7600 nM T82393 CNL60Z 10530046 IC50 = 9.7 nM T82393 C7EU2K 10550226 IC50 = 1 nM T82393 C87ETK 10572102 IC50 = 2.8 nM T82393 CTQ14W 10577036 IC50 = 2800 nM T82393 CD4P1Q 10600659 IC50 = 11000 nM T82393 CL4UB6 10600908 IC50 = 0.61 nM T82393 C1O0FH 10601106 IC50 = 0.79 nM T82393 CCK05R 10601691 IC50 = 6600 nM T82393 C02RNF 10602071 IC50 = 4.2 nM T82393 CZ7QK1 10602072 IC50 = 440 nM T82393 C2YO5H 10602511 IC50 = 1 nM T82393 CW1DA5 10621015 IC50 = 3.4 nM T82393 CY7K4V 10622714 IC50 = 9 nM T82393 CEO5Y7 10648271 IC50 = 1.5 nM T82393 CM4JF2 10649665 IC50 = 3.1 nM T82393 CDH4N3 10666316 IC50 = 1.6 nM T82393 C48GWR 10673548 IC50 = 1.2 nM T82393 CT30EX 10673661 IC50 = 2.8 nM T82393 CWS4N1 10695749 IC50 = 0.23 nM T82393 CE0J9F 10696570 IC50 = 17 nM T82393 COWL53 10696802 IC50 = 0.44 nM T82393 CFE46O 10698171 IC50 = 10 nM T82393 CX6J9R 10719196 IC50 = 2.1 nM T82393 C31LJE 10719273 IC50 = 1.1 nM T82393 CA21RP 10744535 IC50 = 0.66 nM T82393 CJ0KT5 10745306 IC50 = 3000 nM T82393 C3JF9S 10770060 IC50 = 85 nM T82393 CX5Q4G 10787619 IC50 = 1600 nM T82393 CF6X8Z 10792259 IC50 = 1.3 nM T82393 CG6L4E 10814310 IC50 = 0.4 nM T82393 CYO8S1 10837188 IC50 = 3300 nM T82393 C4RWT0 10839079 IC50 = 1.3 nM T82393 C6SDH4 10840060 IC50 = 4500 nM T82393 C6ZSP8 10862104 Ki = 705 nM T82393 CQ1L7C 10863755 Ki = 81 nM T82393 CI7VT4 10864327 IC50 = 400 nM T82393 CF72UK 10864417 IC50 = 12 nM T82393 C6CD3R 10873386 IC50 = 1000 nM T82393 C0AQL8 10873958 Ki = 758 nM T82393 C03WXB 10874655 IC50 = 500 nM T82393 CN75HA 10875139 IC50 = 110 nM T82393 CZ4P3I 10875225 IC50 = 160 nM T82393 CP86EF 10875418 IC50 = 130 nM T82393 CXGN38 10875470 IC50 = 9 nM T82393 CIB8Y1 10884337 Ki = 11 nM T82393 CH3O6X 10886241 IC50 = 190 nM T82393 CG1I4Y 10886343 IC50 = 506 nM T82393 C7V9UQ 10886557 IC50 = 480 nM T82393 CA64PN 10886607 IC50 = 6 nM T82393 C0R5QL 10894433 Ki = 7.15 nM T82393 C7AMS4 10895808 Ki = 153 nM T82393 C10YKE 10896417 IC50 = 200 nM T82393 C24OKB 10896969 IC50 = 300 nM T82393 CMV89R 10897017 IC50 = 6 nM T82393 C3FQT7 10903871 IC50 = 13000 nM T82393 C4EK1H 10907401 IC50 = 140 nM T82393 CSK87I 10907725 IC50 = 42 nM T82393 C69ZTR 10913644 Ki = 3100 nM T82393 C2QR0W 10914151 IC50 = 1000 nM T82393 C2M4PK 10916140 Ki > 780 nM T82393 C7XE3L 10917417 Ki > 1000 nM T82393 C7NS3Y 10917835 IC50 = 2000 nM T82393 CYM85Z 10918704 IC50 = 130 nM T82393 CLIR35 10938505 IC50 = 848 nM T82393 CLOP09 10939716 IC50 = 400 nM T82393 C3EHJ8 10939842 IC50 = 420 nM T82393 CL64UM 10940712 IC50 = 35 nM T82393 C89IYC 10948209 IC50 = 185 nM T82393 C7GH8P 10948665 IC50 = 2700 nM T82393 C2TA9N 10949166 Ki = 7.15 nM T82393 C7PX8G 10960109 Ki > 780 nM T82393 C5HS4F 10961382 Ki = 27 nM T82393 C89LNB 10961787 IC50 = 280 nM T82393 CW17SE 10962269 IC50 = 2200 nM T82393 C0PX9L 10962823 IC50 = 300 nM T82393 C30FBA 10970628 IC50 = 4 nM T82393 CR4QA6 10972932 IC50 = 260 nM T82393 CI34RQ 10973015 IC50 = 550 nM T82393 CA2HJ3 10973131 IC50 = 300 nM T82393 CHL9Z6 10973700 IC50 = 150 nM T82393 C9DM0P 10980832 Ki = 89 nM T82393 CL7K8S 10983560 IC50 = 1400 nM T82393 C3UH2B 10983665 Ki = 10 nM T82393 CJ8I9G 10983916 IC50 = 7 nM T82393 C0ZC7J 10984292 IC50 = 400 nM T82393 C8XD1S 10984566 IC50 = 700 nM T82393 C3FG8K 10984686 IC50 = 490 nM T82393 C5KFS3 10984940 IC50 = 930 nM T82393 C0NIX9 10985227 IC50 = 11 nM T82393 CW8Z6R 10993677 Ki > 1000 nM T82393 CU4TJ5 10994673 IC50 = 0.54 nM T82393 CML07X 10995208 IC50 = 200 nM T82393 CA5I7L 10995373 IC50 = 8 nM T82393 CUAX54 11005498 IC50 = 200 nM T82393 C5JE9G 11014504 IC50 = 160 nM T82393 C8ERT5 11014626 Ki > 780 nM T82393 CO6C8A 11017232 IC50 = 9 nM T82393 CM1H5P 11026185 IC50 = 1000 nM T82393 C5FTO2 11027103 IC50 = 120 nM T82393 CX5FS6 11027381 IC50 = 740 nM T82393 C3LF1Y 11027584 Ki = 51 nM T82393 C8O4VK 11027766 IC50 = 200 nM T82393 C6SA1O 11027809 IC50 = 820 nM T82393 C83AKP 11038896 IC50 = 7.9 nM T82393 CG3B5N 11039339 IC50 = 5 nM T82393 C5R7JX 11049650 Ki = 177 nM T82393 CA85VF 11049836 IC50 = 280 nM T82393 CYA27S 11059553 IC50 = 3700 nM T82393 CH8O1E 11060081 Ki = 17 nM T82393 C49PNL 11069047 IC50 = 1600 nM T82393 C7CH4I 11071209 IC50 = 390 nM T82393 C6EMK9 11071908 IC50 = 94 nM T82393 C3M1JT 11072099 IC50 = 70 nM T82393 C2LSU0 11072397 IC50 = 16 nM T82393 C4OF7J 11080562 IC50 = 700 nM T82393 C7VKE3 11080910 IC50 = 8000 nM T82393 CT3VX4 11080936 Ki = 290 nM T82393 CVJX34 11081788 IC50 = 1300 nM T82393 C6XI8J 11082293 IC50 = 49 nM T82393 C51PQJ 11082573 IC50 = 70 nM T82393 C7N4DG 11082628 IC50 = 600 nM T82393 CUNM68 11083152 Ki = 31 nM T82393 CLFV47 11091348 IC50 = 2500 nM T82393 C3S6TD 11091368 IC50 > 50000 nM T82393 COZ9U1 11092188 IC50 = 700 nM T82393 CL7R9U 11092806 IC50 = 460 nM T82393 C6R7XB 11092861 Ki = 242 nM T82393 CWT6C7 11092884 IC50 = 8 nM T82393 C6CLV8 11101735 IC50 = 942 nM T82393 C57OXT 11102540 IC50 = 310 nM T82393 CA2OS3 11103408 IC50 = 5 nM T82393 CGE45I 11103515 IC50 = 200 nM T82393 CFA08I 11103765 IC50 = 220 nM T82393 C2QS0G 11103972 IC50 = 130 nM T82393 C6G2DI 11111616 Ki = 734 nM T82393 CWV45Z 11112302 Ki = 621 nM T82393 CEAI92 11112993 IC50 = 416 nM T82393 C14PKX 11113492 IC50 = 680 nM T82393 CD57BU 11113544 IC50 = 4490 nM T82393 C8HIY0 11113868 IC50 = 200 nM T82393 CI1GS5 11114351 IC50 = 22 nM T82393 CUO7B3 11122933 IC50 = 2400 nM T82393 C60PHT 11124083 IC50 = 300 nM T82393 CU8VN1 11124523 IC50 = 120 nM T82393 CE28RK 11124637 IC50 = 580 nM T82393 C3PR1J 11124862 IC50 = 14 nM T82393 CAJ27B 11124943 IC50 = 8 nM T82393 C9GJ7C 11133809 Ki > 10010 nM T82393 CU2C9O 11135818 IC50 = 180 nM T82393 C3PZ0C 11135829 IC50 = 120 nM T82393 CPO02F 11142863 IC50 = 177 nM T82393 C8HM2R 11145437 Ki = 56 nM T82393 C0ACW4 11146109 IC50 = 1170 nM T82393 CD9HN2 11146249 IC50 = 1000 nM T82393 CHF19X 11146467 Ki = 77 nM T82393 CVI3F8 11188429 IC50 = 201 nM T82393 CO5VN2 11201367 IC50 = 54 nM T82393 CET3R7 11201814 IC50 = 134 nM T82393 C43ONW 11202395 IC50 = 9 nM T82393 C72UCB 11233687 IC50 = 94 nM T82393 CPV9L7 11246575 Ki = 0.53 nM T82393 CH6E8G 11247057 IC50 = 80 nM T82393 CJZ3P6 11257884 Ki > 1000 nM T82393 CD1FT8 11258906 IC50 = 69 nM T82393 CC62RY 11279665 IC50 = 15 nM T82393 CP17ID 11284983 IC50 = 34000 nM T82393 C1IW7N 11292680 IC50 = 14000 nM T82393 C8C5AV 11294179 IC50 = 130 nM T82393 CQH57S 11342435 IC50 > 25000 nM T82393 CCKI02 11360440 Ki = 15 nM T82393 C48DYJ 11374008 Ki = 1.7 nM T82393 CL8QO7 11382562 IC50 = 4 nM T82393 CNZ0T5 11386918 IC50 = 72 nM T82393 C9KVB7 11394505 IC50 = 24 nM T82393 C9ABX8 11397130 IC50 = 1600 nM T82393 C3EX5J 11407165 Ki = 21 nM T82393 C2EUO5 11417011 IC50 = 50 nM T82393 C5NAJ3 11449819 IC50 = 30 nM T82393 C5QEZ8 11483818 IC50 = 375 nM T82393 C9QW0X 11497618 IC50 = 890 nM T82393 C9DSV5 11502876 IC50 = 2960 nM T82393 C6K2JL 11509086 Ki = 238 nM T82393 CWS35C 11510523 IC50 = 140 nM T82393 C5VUM2 11517085 Ki = 160 nM T82393 CX0B1M 11524708 IC50 = 1430 nM T82393 C6OXQ8 11524821 Ki = 41 nM T82393 CGC73J 11531219 Ki = 188 nM T82393 C9Y6LH 11533683 IC50 = 370 nM T82393 CV19DJ 11533863 IC50 = 1180 nM T82393 CBQ80H 11546305 Ki = 8 nM T82393 CLY2P6 11552350 Ki = 391 nM T82393 C3FW5A 11554783 IC50 = 1710 nM T82393 CI4Z0L 11560876 Ki = 323 nM T82393 CGK97A 11560983 IC50 = 1610 nM T82393 C0M5KB 11563197 IC50 = 2300 nM T82393 CPHL63 11566516 Ki = 6 nM T82393 C5NOF7 11566672 Ki = 66 nM T82393 CQ58KF 11567255 Ki = 96 nM T82393 C5WBJ4 11568227 Ki = 400 nM T82393 CVCJ29 11570382 IC50 = 1250 nM T82393 CRJY76 11575575 IC50 = 1560 nM T82393 CHV2G1 11575995 Ki = 4 nM T82393 CW62GP 11576985 IC50 = 2150 nM T82393 CH6WQ5 11584432 IC50 = 1900 nM T82393 C34HSK 11591268 IC50 = 630 nM T82393 CTQ87G 11599024 IC50 = 80 nM T82393 CVGC49 11603611 Ki = 5 nM T82393 C6M2NF 11606412 IC50 = 2240 nM T82393 C81DCM 11606523 IC50 = 980 nM T82393 CJ0TZ5 11613968 IC50 = 970 nM T82393 C3JO7H 11627426 IC50 = 1230 nM T82393 CXC8K6 11630678 Ki = 28 nM T82393 CCBS59 11634234 IC50 = 1.5 nM T82393 C8UMG3 11634941 IC50 = 3590 nM T82393 CR1OZ4 11639207 Ki = 100 nM T82393 CNY92D 11640694 Ki = 400 nM T82393 C64JZH 11646633 Ki = 53 nM T82393 CDB94C 11648703 IC50 = 2310 nM T82393 CU1W8B 11653224 Ki = 3 nM T82393 CPJ8K9 11663500 IC50 = 0.9 nM T82393 C94GZV 11664224 IC50 = 1500 nM T82393 CK2G8Y 11667693 Ki = 943 nM T82393 CR68FB 11668295 Ki = 5.5 nM T82393 C86PCY 11668526 Ki = 1440 nM T82393 C0FT5I 11671315 IC50 = 2240 nM T82393 C6D1FB 11674794 Ki = 800 nM T82393 CK0QJ7 11675173 Ki = 7 nM T82393 C57TOX 11676244 IC50 = 280 nM T82393 C0C6NY 11682301 Ki = 487 nM T82393 C1S7CM 11683254 Ki = 755 nM T82393 C7GX2W 11695181 Ki = 209 nM T82393 C3U6ZR 11697504 Ki = 11 nM T82393 CY6E3B 11697569 IC50 = 1570 nM T82393 C4BGI2 11698938 IC50 = 1 nM T82393 CS28MX 11704287 IC50 = 2530 nM T82393 C07CWS 11710815 Ki = 456 nM T82393 CT8U3E 11711300 IC50 = 8200 nM T82393 C2PG8W 11713566 IC50 = 3450 nM T82393 CWL6A1 11713901 IC50 = 4400 nM T82393 C2BJ3X 11716217 Ki = 23 nM T82393 C2NVO9 11717506 Ki = 764 nM T82393 CBUA07 11729454 IC50 = 2.25 nM T82393 C9J5VX 11730465 IC50 = 700 nM T82393 CJ31ZC 11730692 IC50 = 500 nM T82393 C3H4NC 11730693 IC50 = 490 nM T82393 CBT48P 11731926 Ki = 13.7 nM T82393 CA43HK 11732287 IC50 = 180 nM T82393 C68KBY 11732585 Ki = 129 nM T82393 CRA40L 11733697 IC50 = 500 nM T82393 C64LQC 11733862 IC50 = 2 nM T82393 C27SBC 11734162 IC50 = 492 nM T82393 CIU03K 11734219 Ki = 10 nM T82393 C6HV8Z 11752434 IC50 = 19 nM T82393 CO8QT0 11753905 IC50 = 0.14 nM T82393 CF2J8V 11758099 IC50 = 39.81 nM T82393 C3RW1X 11761191 IC50 = 3800 nM T82393 C6K8HR 11761578 Ki = 229 nM T82393 CE1HZ4 11761760 IC50 = 2300 nM T82393 C04DFH 11783486 Ki = 4.9 nM T82393 CRA5H1 11793654 IC50 = 13 nM T82393 CU7M8D 11793896 IC50 = 1.5 nM T82393 C6X3PH 11798586 IC50 = 6700 nM T82393 C62FGK 11799105 IC50 = 9.5 nM T82393 C8HA3G 11799315 IC50 = 4900 nM T82393 C3OJS7 11799603 IC50 = 1.25 nM T82393 CC3MQ4 11813457 IC50 = 200 nM T82393 CZ08ID 11814382 IC50 = 6 nM T82393 CEN02U 11822212 Ki = 484 nM T82393 CDU9S2 11824087 Ki = 71 nM T82393 C3VO5H 11824148 Ki = 12.9 nM T82393 C23WZY 11824787 IC50 = 5.9 nM T82393 C7BK5P 11825105 IC50 = 805 nM T82393 C57LPO 11826993 IC50 = 980 nM T82393 CDOR01 11827696 IC50 = 270 nM T82393 C48QEH 11833533 Ki = 391 nM T82393 CR3WH6 11854559 IC50 = 0.6 nM T82393 CNT08B 11854813 IC50 = 1 nM T82393 C2PW6M 11854816 IC50 = 2.512 nM T82393 CYKX65 11854817 IC50 = 0.6 nM T82393 CZDB06 11855066 IC50 = 0.631 nM T82393 COEX56 11855067 IC50 = 0.6 nM T82393 CKB41C 11855068 IC50 = 1 nM T82393 CKTG95 11855069 IC50 = 0.6 nM T82393 CT8AX3 11855070 IC50 = 4.7 nM T82393 C0V7WA 11855071 IC50 = 1.259 nM T82393 CSX7Y9 11855326 IC50 = 0.7943 nM T82393 C4WNG0 11855327 IC50 = 7.943 nM T82393 CLS41N 11855328 IC50 = 0.631 nM T82393 CA9Y5M 11855329 IC50 = 1.259 nM T82393 CNU37H 11855330 IC50 = 0.5012 nM T82393 CM93GN 11855331 IC50 = 0.7943 nM T82393 CDNK35 11855595 IC50 = 0.631 nM T82393 CN3Y4O 11855596 IC50 = 3.162 nM T82393 CSB18V 11855599 IC50 = 1.259 nM T82393 CK5S0D 11855600 IC50 = 1.3 nM T82393 CG6N1F 11856141 IC50 = 0.5 nM T82393 C6L8YM 11856142 IC50 = 6.2 nM T82393 CFL1S4 11856418 IC50 = 0.3981 nM T82393 C86VAX 11856419 IC50 = 0.6 nM T82393 CYDS54 11856677 IC50 = 0.6 nM T82393 CENK97 11856678 IC50 = 2.3 nM T82393 CX7K1N 11856679 IC50 = 9.6 nM T82393 C9GD2X 11856681 IC50 = 100 nM T82393 C2ANV3 11856682 IC50 = 0.6 nM T82393 CBD01L 11856948 IC50 = 1.259 nM T82393 C4XR5G 11963536 IC50 = 2.2 nM T82393 CB80OT 12000718 IC50 > 20000 nM T82393 C43PJZ 12000720 IC50 > 20000 nM T82393 C70TDZ 15503645 IC50 = 47 nM T82393 C47RXG 15541745 IC50 = 9 nM T82393 CEFV16 15541746 IC50 = 58000 nM T82393 C1GW2T 15541747 IC50 = 6 nM T82393 CU05VE 15541748 IC50 = 18 nM T82393 CU7CM3 15551877 IC50 = 277 nM T82393 CO2XY0 15851477 IC50 = 2 nM T82393 CY0S2M 15851478 IC50 = 0.8 nM T82393 C6R1LD 15985818 IC50 = 2 nM T82393 CR95VN 15986108 IC50 = 32.82 nM T82393 C2PF7G 15986113 IC50 = 0.5 nM T82393 CNX86Z 15986115 IC50 = 920 nM T82393 CH3YK2 15986256 IC50 = 0.66 nM T82393 CS4T2X 15986257 IC50 = 0.53 nM T82393 CV67UL 15986261 IC50 = 60 nM T82393 CM04UZ 15986512 IC50 = 1500 nM T82393 C8XK3C 15986607 IC50 = 1.04 nM T82393 COQ05K 15986703 IC50 = 1.07 nM T82393 C9N0JM 15986869 IC50 = 320 nM T82393 C6KR4A 15986873 IC50 = 230 nM T82393 CU2C1R 15987326 IC50 = 3 nM T82393 C15LJN 15987412 IC50 = 30 nM T82393 CUQG04 16130642 IC50 = 4453 nM T82393 CQS0F5 16719301 IC50 > 10000 nM T82393 C75XDI 16730519 IC50 = 130 nM T82393 C2W1VA 16739287 Ki = 28 nM T82393 CZ1EY7 17754304 Ki = 0.26 nM T82393 C3S2TQ 17754305 Ki = 0.62 nM T82393 CXCJ91 17754605 Ki = 0.52 nM T82393 C49QVS 17754779 Ki = 0.2 nM T82393 CSV68X 17754781 Ki = 0.06 nM T82393 CIR7S8 17866387 IC50 = 108 nM T82393 CL1H9W 17866459 IC50 = 146 nM T82393 C9RNH3 17866675 IC50 = 154 nM T82393 CCGR13 17897285 IC50 = 203 nM T82393 C2ZAX1 18002715 IC50 = 190 nM T82393 C12UGK 18002722 IC50 = 160 nM T82393 C0IYW8 18002726 IC50 = 230 nM T82393 C8N1DM 18002729 IC50 = 240 nM T82393 CCG96A 18002736 IC50 = 83 nM T82393 C5MLG1 18002745 IC50 = 510 nM T82393 CXT4H2 18002752 IC50 > 3000 nM T82393 C26WHK 18002758 IC50 = 1 nM T82393 CV90XS 18002764 IC50 = 250 nM T82393 C8KPM7 18002765 IC50 > 1000 nM T82393 CMJ0K3 18002771 IC50 = 250 nM T82393 C2CO9Z 18002775 IC50 = 900 nM T82393 CM48NU 18324856 IC50 = 4 nM T82393 CI53DY 18379040 IC50 = 119 nM T82393 CB1U5T 18379077 IC50 = 490 nM T82393 C3LPD2 18379087 IC50 > 3000 nM T82393 CSX97G 18379115 IC50 = 45 nM T82393 CJHL25 18379123 IC50 = 143 nM T82393 CR0B8G 18379149 IC50 = 737 nM T82393 CS4V5K 18379187 IC50 = 56 nM T82393 CCTY94 18379210 IC50 = 290 nM T82393 CA6K5S 18379235 IC50 = 89 nM T82393 CCSK49 18379254 IC50 = 30 nM T82393 CP4T7S 18379435 IC50 = 105 nM T82393 C30EAU 20651317 IC50 = 4 nM T82393 C48TWB 20728102 IC50 = 560 nM T82393 C0B7VU 20748471 Ki = 1200 nM T82393 C92BJM 20748508 Ki = 360 nM T82393 C91SKR 20748648 Ki = 20000 nM T82393 CZ9G3R 20748736 Ki = 190 nM T82393 CWP27B 20748738 Ki = 4000 nM T82393 CM92DX 21304705 IC50 = 28 nM T82393 CJ0Y9V 21304706 IC50 = 40 nM T82393 C5X1YM 21304708 IC50 = 42 nM T82393 C0Z3LD 21304710 IC50 = 19 nM T82393 CG18HB 21310751 IC50 = 218 nM T82393 CEW0M3 21310753 IC50 = 243 nM T82393 CC2L1Z 21310756 IC50 = 429 nM T82393 C0T2QX 21310757 IC50 = 173 nM T82393 C5SG2L 21310789 IC50 = 210 nM T82393 C3TI6Y 21310790 IC50 = 61 nM T82393 C87BMF 21310824 IC50 = 174 nM T82393 C26IPQ 21310829 IC50 = 70 nM T82393 CIB1X5 21310851 IC50 = 157 nM T82393 CUJ6A1 21310984 IC50 = 377 nM T82393 CH6U1G 22338710 IC50 = 467 nM T82393 CO91AD 22341241 IC50 = 150 nM T82393 C9BT5F 22626996 IC50 = 2.1 nM T82393 C7ITG0 22644780 IC50 = 23 nM T82393 CIQ76F 22644837 IC50 = 74 nM T82393 CYJ48I 22644895 IC50 = 20 nM T82393 CQB36V 22644965 IC50 = 10 nM T82393 CVM1O6 22644970 IC50 = 83 nM T82393 C0K1GE 22645081 IC50 = 7 nM T82393 CF75MS 23017979 IC50 = 2.2 nM T82393 CQJ3S4 23018008 IC50 = 20 nM T82393 C4VG8C 23506747 IC50 = 122 nM T82393 CK97AT 23506779 IC50 = 67 nM T82393 CP94QR 23506783 IC50 = 32 nM T82393 CM5Z8D 23513782 IC50 = 2.5 nM T82393 CX32YK 23513795 IC50 < 1 nM T82393 C6IZ1S 23513821 IC50 = 3.4 nM T82393 CPNM93 23513825 IC50 = 1 nM T82393 CML90Q 23513831 IC50 = 2.2 nM T82393 C87RTM 23513845 IC50 = 4.8 nM T82393 CNSU58 23513850 IC50 = 2 nM T82393 C4R2AJ 23625454 IC50 = 3600 nM T82393 CD3U8A 23627203 Ki = 10 nM T82393 CL24JR 23655078 IC50 = 3 nM T82393 CG3J2L 24768528 IC50 = 1.6 nM T82393 C80UHK 24799267 Ki = 1100 nM T82393 C5M9JF 24799268 Ki = 70 nM T82393 CE4O5B 24799438 Ki = 80 nM T82393 C0R1XH 24799439 Ki = 3000 nM T82393 CXA42B 24799440 Ki = 70 nM T82393 CS65UC 24799441 Ki = 240 nM T82393 C3VWC9 24799442 Ki = 140 nM T82393 C92PBT 24799443 Ki = 16 nM T82393 CB1T2S 24799616 Ki = 5 nM T82393 C20YMK 24799617 Ki = 100 nM T82393 CZMO02 24799618 Ki = 2700 nM T82393 C1DO9Y 24799619 Ki = 11 nM T82393 C4L0EV 24799620 Ki = 3000 nM T82393 CMBT43 24799621 Ki = 9 nM T82393 C2KPS9 24799777 Ki = 5000 nM T82393 C5M3YW 24799779 Ki = 3 nM T82393 CO3J8Y 24799780 Ki = 14 nM T82393 C0YJ1H 24799781 Ki = 1 nM T82393 CS0C5J 24799782 Ki = 130 nM T82393 CW3A9R 24799951 Ki = 260 nM T82393 CYG49P 24799952 Ki > 100000 nM T82393 CX6A5S 24799953 Ki > 100000 nM T82393 C2D5PK 24799954 Ki = 3100 nM T82393 CU2YV9 24799955 Ki = 26000 nM T82393 CZ5TW6 24799956 Ki = 420 nM T82393 CL0WA5 24799957 Ki = 80 nM T82393 CMRD73 24800654 Ki = 12 nM T82393 C5TD9X 24800829 Ki = 700 nM T82393 C7TZ4K 24800833 Ki = 8 nM T82393 CYD3F8 24801010 Ki = 11 nM T82393 C1SCD0 24801011 Ki = 8 nM T82393 CEG51N 24801012 Ki = 140 nM T82393 CAF90P 24801013 Ki = 3000 nM T82393 CG76XQ 24801014 Ki = 110 nM T82393 CI69GF 24801015 Ki = 18 nM T82393 C18FRG 24807817 IC50 > 100000 nM T82393 C9L6VE 24860419 Ki = 800 nM T82393 C4LXM8 24860420 IC50 = 3.3 nM T82393 CK0CI6 24860421 IC50 = 10 nM T82393 C4SL8W 24860422 IC50 = 64.5 nM T82393 CZI59C 24860423 IC50 = 2 nM T82393 CE29HI 24860424 IC50 = 6.4 nM T82393 CT10JE 24860425 IC50 < 1 nM T82393 CRC98J 24860426 IC50 = 2.5 nM T82393 C8MKR0 24860427 IC50 = 3.5 nM T82393 C3S6DX 24860428 IC50 = 3500 nM T82393 C2LNE4 24860429 IC50 = 4 nM T82393 CF4D0X 24860430 IC50 = 27 nM T82393 C0G8KH 24873166 Ki = 4818 nM T82393 CY0A9K 24873286 Ki = 5 nM T82393 C3U8ZQ 24882385 IC50 = 60 nM T82393 C1M9QW 24888678 Ki = 10 nM T82393 CH8PQ0 24890899 Ki = 2 nM T82393 C2FI5D 24978491 Ki = 0.18 nM T82393 CNCA57 25004194 Ki > 1000 nM T82393 CA5DJ4 25138228 Ki = 0.14 nM T82393 C51TNU 25138229 Ki = 6.7 nM T82393 C9HVG2 25138230 Ki = 30 nM T82393 CKLM60 25138231 Ki = 32 nM T82393 CT2B8V 25138232 Ki = 32 nM T82393 C2G8QJ 25138233 Ki = 33 nM T82393 CN8V7O 25138234 Ki = 53 nM T82393 C6PR5O 25138235 Ki = 137 nM T82393 C6Z3VR 25138236 Ki = 40 nM T82393 C3PL2Y 25138237 Ki = 94 nM T82393 CT3NV5 25138238 Ki = 143 nM T82393 CF1W2Q 25138239 Ki = 673 nM T82393 C3B7GM 25138240 Ki = 2140 nM T82393 C01VIC 25138241 Ki = 3070 nM T82393 CM3Q7D 25138242 Ki = 3220 nM T82393 C1C2YR 25138243 Ki > 50000 nM T82393 C8R2WY 25138244 Ki = 13 nM T82393 CX6D9J 25138245 Ki = 55 nM T82393 CSK09Y 25138246 Ki = 530 nM T82393 CLJ9N1 25138247 Ki = 3400 nM T82393 C5RG9J 25138248 Ki = 11 nM T82393 CPM9C1 25138249 Ki = 5 nM T82393 C7A6JQ 25138250 Ki = 52 nM T82393 CAE20Q 25138251 Ki = 27 nM T82393 CUT69K 25138252 Ki = 8 nM T82393 C3RA1L 25138253 Ki = 2 nM T82393 C4T6DU 25138254 Ki = 4.5 nM T82393 CC0LB7 25138255 Ki = 50 nM T82393 CB7V8Y 25147773 IC50 = 55 nM T82393 CEP9Q2 25180867 IC50 = 2290 nM T82393 CHR2P1 25183768 Ki > 25000 nM T82393 C0H3RD 42627769 IC50 = 140 nM T82393 CPO1Z3 44123600 IC50 > 1000 nM T82393 C25ELB 44143088 IC50 = 74131.02 nM T82393 CWS64Q 44143474 IC50 = 33 nM T82393 C7HV5Q 44143475 IC50 = 1 nM T82393 C06IJY 44143476 IC50 = 2 nM T82393 CVM82U 44143477 IC50 = 2 nM T82393 C5XEB8 44143478 IC50 = 1 nM T82393 CJQF59 44143479 IC50 = 73 nM T82393 C0ZW7S 44143480 IC50 = 2 nM T82393 C7K0YS 44143481 IC50 < 1 nM T82393 CWU1K0 44143482 IC50 = 2 nM T82393 CA29EQ 44143483 IC50 = 3 nM T82393 CA5P3E 44143484 IC50 = 11 nM T82393 C7ER1N 44143485 IC50 = 9 nM T82393 C8YNO3 44143486 IC50 = 65 nM T82393 CLJG93 44143487 IC50 = 1.2 nM T82393 CJB54F 44143488 IC50 = 10 nM T82393 CT80ED 44219901 IC50 = 35000 nM T82393 C9T5ZF 44220093 IC50 > 100000 nM T82393 CCI64J 44224245 IC50 = 40000 nM T82393 C5S6QR 44253975 IC50 = 28600 nM T82393 CN9BZ7 44253976 IC50 = 2230 nM T82393 CTX92S 44272249 IC50 = 28 nM T82393 CG92WS 44272353 IC50 = 25 nM T82393 C3KY9R 44272354 IC50 = 27 nM T82393 C43QPI 44272355 IC50 = 84 nM T82393 CVM59X 44272455 IC50 = 28 nM T82393 CO2Z6K 44272475 IC50 = 26 nM T82393 C63KSL 44272540 IC50 = 42 nM T82393 CTO6V2 44278377 IC50 = 5 nM T82393 C1K6CY 44278395 IC50 = 11 nM T82393 CG2HL4 44278396 IC50 = 10 nM T82393 C2Z6MF 44278411 IC50 = 67 nM T82393 C9X8DM 44278412 IC50 = 10 nM T82393 CJ8ON1 44278424 IC50 = 21 nM T82393 CEA0H3 44278449 IC50 = 8 nM T82393 C5ZGQ9 44278455 IC50 = 49 nM T82393 CC4V8G 44278484 IC50 = 7 nM T82393 CDGF86 44278511 IC50 = 67 nM T82393 CJ78PR 44278512 IC50 = 15 nM T82393 C1GLP0 44278522 IC50 = 15 nM T82393 CAB1C5 44278523 IC50 = 28000 nM T82393 C04WHR 44278532 IC50 = 77000 nM T82393 CK16OS 44278550 IC50 = 27 nM T82393 CJ94UF 44278576 IC50 = 120 nM T82393 CQDI85 44278667 IC50 = 9600 nM T82393 CLT4A9 44278705 IC50 = 7 nM T82393 C6S3GN 44283598 IC50 = 205 nM T82393 CXE73H 44283613 IC50 = 86 nM T82393 CP3L2U 44283938 IC50 > 1000 nM T82393 C3UB9V 44286654 Ki = 1.85 nM T82393 CB07MX 44286663 Ki = 0.84 nM T82393 C3KXY9 44286674 Ki = 1.85 nM T82393 C4LI6F 44293416 IC50 = 1800 nM T82393 CAFB18 44296974 Ki = 544 nM T82393 CALD50 44304020 IC50 > 10000 nM T82393 CTU4S6 44304048 IC50 > 3000 nM T82393 C7L9JK 44304111 Ki = 10 nM T82393 C0IJ9D 44304112 Ki = 27.6 nM T82393 CSVK45 44304230 IC50 > 10000 nM T82393 CJ53NI 44304355 IC50 = 76 nM T82393 C5QUK2 44308295 Ki = 64 nM T82393 C2E4IT 44308297 Ki = 27 nM T82393 C0K4UQ 44308298 Ki = 20 nM T82393 CCRW50 44308304 Ki = 55 nM T82393 CZF5S2 44308327 Ki = 29 nM T82393 COE56H 44308377 Ki = 142 nM T82393 C7OT6S 44308488 Ki = 156 nM T82393 CI2Z0H 44308525 Ki = 16 nM T82393 CU0J5A 44308623 Ki = 31 nM T82393 CSEB94 44308624 Ki = 11 nM T82393 CST39W 44308640 Ki = 20 nM T82393 C4SJF3 44309329 IC50 = 194 nM T82393 C7ED1H 44309330 IC50 = 294 nM T82393 C1E3KF 44309437 IC50 = 64 nM T82393 CH3SU2 44309482 IC50 = 285 nM T82393 CQ7Z0W 44309533 IC50 = 57 nM T82393 CJ0L4P 44309550 IC50 = 727 nM T82393 C0WIG9 44309577 IC50 = 28 nM T82393 C6J3WN 44309662 IC50 = 133 nM T82393 C49MHR 44309863 IC50 = 23 nM T82393 CMW0U4 44309879 IC50 = 633 nM T82393 CK6BT0 44309901 IC50 = 56 nM T82393 C0HR5Q 44316157 IC50 = 38 nM T82393 CSA5P7 44316333 IC50 = 81 nM T82393 CS7D5E 44317086 IC50 = 39 nM T82393 C8JW4D 44322861 IC50 = 830 nM T82393 CQK83T 44322917 IC50 = 1510 nM T82393 CQ4P7G 44322988 IC50 = 85 nM T82393 CT9P2I 44322993 IC50 = 300 nM T82393 C6UFO3 44323025 IC50 = 83 nM T82393 CDK3O7 44323042 IC50 = 100 nM T82393 CF0H4O 44323043 IC50 = 150 nM T82393 C0UY1E 44323088 IC50 = 170 nM T82393 C15SKA 44323114 IC50 = 690 nM T82393 C4DAP9 44323115 IC50 = 210 nM T82393 CGO78N 44323126 IC50 = 100 nM T82393 CXUF49 44323141 IC50 = 760 nM T82393 CA50CN 44323145 IC50 = 270 nM T82393 CF65YI 44323249 IC50 = 950 nM T82393 CPX1B7 44323277 IC50 = 850 nM T82393 CO67AU 44323310 IC50 = 1200 nM T82393 CO0S9J 44325072 Ki = 67 nM T82393 C4R9LM 44325085 Ki = 1.6 nM T82393 CL8MD0 44325156 Ki = 8.7 nM T82393 CV3S9G 44325157 Ki = 340 nM T82393 C9MD1A 44325159 Ki = 510 nM T82393 C6R4NI 44325225 Ki = 22 nM T82393 C3M2XY 44325277 Ki = 71 nM T82393 CA4FQ5 44325443 Ki = 21 nM T82393 C2ZH0F 44327181 IC50 = 4 nM T82393 C8V3AO 44327386 IC50 = 17 nM T82393 C0UC5H 44327407 IC50 = 10 nM T82393 C6TPB1 44327409 IC50 = 6 nM T82393 C8ZI0P 44327432 IC50 = 18 nM T82393 CVJ9Q6 44327443 IC50 = 5 nM T82393 C4R9WM 44327681 IC50 = 26 nM T82393 C6IM7G 44327755 IC50 = 3 nM T82393 CHU2P7 44328876 IC50 = 157 nM T82393 C0KA4S 44328937 IC50 = 69 nM T82393 CLT8B6 44328971 IC50 = 254 nM T82393 C7J0ZI 44329016 IC50 = 157 nM T82393 CW24VN 44329040 IC50 = 528 nM T82393 C9J0VO 44329253 IC50 = 157 nM T82393 C3YAF6 44329898 IC50 = 3 nM T82393 C2K6OU 44329943 IC50 = 199.53 nM T82393 C5BYR4 44329998 IC50 = 180 nM T82393 C0SMC9 44330092 IC50 = 1.5 nM T82393 C35SIO 44330094 IC50 = 6.31 nM T82393 C3NM2G 44330095 IC50 = 2.512 nM T82393 C6SCU5 44330119 IC50 = 3.162 nM T82393 C69KPL 44330130 IC50 = 7.943 nM T82393 C9P6ZF 44330131 IC50 = 5.012 nM T82393 C9R1ZE 44330132 IC50 = 3 nM T82393 CKS01F 44330133 IC50 = 31.62 nM T82393 CLU8I7 44330135 IC50 = 15 nM T82393 C1IE0S 44330147 IC50 = 6 nM T82393 CPG7N2 44330149 IC50 = 4.5 nM T82393 CYP6S4 44330152 IC50 = 60 nM T82393 CMGA28 44330163 IC50 = 3.5 nM T82393 CXI49L 44330197 IC50 = 74 nM T82393 CDQM84 44330198 IC50 = 7.9 nM T82393 CH6EN4 44330225 IC50 = 55 nM T82393 C3GA9Q 44330226 IC50 = 6 nM T82393 CD0L6S 44331932 IC50 = 87 nM T82393 CHIG68 44331976 IC50 = 26 nM T82393 CF4JN0 44331983 IC50 = 49 nM T82393 CG2AH4 44331984 IC50 = 210 nM T82393 CPB96A 44332003 IC50 = 200 nM T82393 C6RE3I 44332107 IC50 = 80 nM T82393 C3L1HQ 44332161 IC50 = 63 nM T82393 CY0MQ9 44332313 IC50 = 36 nM T82393 C0Y2CZ 44339375 IC50 = 300 nM T82393 CP12TJ 44339394 IC50 = 1000 nM T82393 C30YNC 44339395 IC50 = 31 nM T82393 COR15M 44339402 IC50 = 25 nM T82393 CU5NI2 44339444 IC50 = 28 nM T82393 CISO73 44339448 IC50 = 5 nM T82393 C4QKI6 44339451 IC50 = 40 nM T82393 CEUP59 44339452 IC50 = 3000 nM T82393 CU7DZ9 44339462 IC50 = 400 nM T82393 CLT8C6 44339543 IC50 = 6 nM T82393 C6M4UR 44339544 IC50 = 2000 nM T82393 C5PQ1B 44339569 IC50 = 7 nM T82393 CA65PF 44339570 IC50 = 6 nM T82393 C4W8LS 44339571 IC50 = 19 nM T82393 COUE24 44339575 IC50 = 7 nM T82393 CE90PW 44339624 IC50 = 68 nM T82393 CMA2L3 44339647 IC50 = 14 nM T82393 CFCZ60 44339648 IC50 = 26 nM T82393 CW8DO2 44339742 IC50 = 32 nM T82393 C3EX8J 44342378 IC50 > 10000 nM T82393 C5XD4N 44363290 IC50 = 22 nM T82393 C52RVU 44363311 IC50 = 4400 nM T82393 CB0GO6 44363331 IC50 = 1.4 nM T82393 C3WXU0 44363479 IC50 = 1.3 nM T82393 C2JGR5 44363482 IC50 = 6100 nM T82393 CT9MR2 44363517 IC50 = 9 nM T82393 CR52AW 44363562 IC50 = 0.21 nM T82393 CKO2D4 44363576 IC50 = 3.3 nM T82393 CT3OG2 44363603 IC50 = 13 nM T82393 CH72OI 44363783 IC50 = 0.8 nM T82393 C68YSD 44363884 IC50 = 6.6 nM T82393 CYE90S 44383704 Ki = 33.2 nM T82393 C4O9DP 44383747 Ki = 7.89 nM T82393 C0W2SV 44383786 Ki = 21.7 nM T82393 C2UNW6 44383789 Ki = 8.92 nM T82393 C6V9FQ 44383801 Ki = 42.2 nM T82393 CV8UX5 44383829 Ki = 13.8 nM T82393 CCY30B 44383847 Ki = 90.2 nM T82393 C7MLD8 44383849 Ki = 15.5 nM T82393 C9F5LS 44384003 Ki = 59.6 nM T82393 CSM3P7 44384004 Ki = 75.8 nM T82393 CO9LJ6 44384005 Ki = 777 nM T82393 CJ4NV9 44384173 Ki = 73.6 nM T82393 C7B3AN 44384343 Ki = 37.4 nM T82393 C4B9NU 44384357 Ki = 22.8 nM T82393 CC81JP 44384395 Ki = 2.2 nM T82393 CKG95Y 44384455 Ki > 780 nM T82393 C96PAY 44384542 Ki = 120 nM T82393 C5ZYN1 44384591 Ki = 500 nM T82393 CVZ42A 44384592 Ki = 37.4 nM T82393 C49TAV 44384649 Ki = 11.2 nM T82393 CALI01 44384650 Ki = 18.9 nM T82393 C8SCB5 44384659 IC50 > 10000 nM T82393 C7A2HC 44384755 Ki = 7.99 nM T82393 CL51XE 44384756 Ki = 6.45 nM T82393 CD2PM4 44384761 Ki = 50 nM T82393 CJH8P4 44384762 Ki = 2.98 nM T82393 C59NBH 44384814 Ki = 32.7 nM T82393 C5AE0O 44384972 Ki = 14.2 nM T82393 CZ6PU7 44389401 Ki > 1000 nM T82393 CO4W0Y 44389552 Ki > 1000 nM T82393 C3YPG6 44390245 IC50 = 19 nM T82393 COG80H 44390258 IC50 = 14 nM T82393 C0U3XR 44390274 IC50 = 35 nM T82393 CAC3F2 44390281 IC50 = 11 nM T82393 CRE9G2 44390289 IC50 = 13 nM T82393 CN41JE 44390299 IC50 = 19 nM T82393 C5VBL2 44390300 IC50 = 23 nM T82393 C4YUK7 44390304 IC50 = 68 nM T82393 C47EZV 44390314 IC50 = 7 nM T82393 CF65OK 44390317 IC50 = 15 nM T82393 CV45JT 44390322 IC50 = 24 nM T82393 C3GU1Q 44390323 IC50 = 61 nM T82393 CAZ2B4 44390326 IC50 = 12 nM T82393 C2Y7MR 44390338 IC50 = 75 nM T82393 CA47CR 44390351 IC50 = 5 nM T82393 CYW89M 44390352 IC50 = 30 nM T82393 CPK9Z6 44390355 IC50 = 28 nM T82393 CEJH75 44390356 IC50 = 37 nM T82393 CWYM93 44390391 IC50 = 10 nM T82393 CMGB67 44393214 IC50 = 69 nM T82393 CA1S5T 44393217 IC50 = 92 nM T82393 CSC6N1 44393218 IC50 = 121 nM T82393 CBO9E6 44393239 IC50 = 130 nM T82393 CQNR83 44393261 IC50 = 49 nM T82393 CT1LM8 44393266 IC50 = 197 nM T82393 C0SGF6 44393279 IC50 = 14 nM T82393 CYFC07 44393295 IC50 = 18 nM T82393 C24INM 44393328 IC50 = 14 nM T82393 C15IZJ 44393358 IC50 = 31 nM T82393 C3HP5Q 44393383 IC50 = 89 nM T82393 CS06PD 44393394 IC50 = 41 nM T82393 CFA83O 44393414 IC50 = 81 nM T82393 CCO3S9 44393444 IC50 = 418 nM T82393 CNO4P6 44393516 IC50 = 180 nM T82393 C5OIK4 44393520 IC50 = 1070 nM T82393 C80NZE 44394179 IC50 = 20 nM T82393 CN7WS6 44394426 IC50 = 7.2 nM T82393 CN6GO3 44394819 IC50 = 15 nM T82393 CVGU01 44394916 IC50 = 8.3 nM T82393 CG1W0V 44394994 IC50 = 33 nM T82393 CT6VX4 44395030 IC50 = 17 nM T82393 C2EG4V 44395069 IC50 = 14 nM T82393 CT5N1F 44395157 IC50 = 2.2 nM T82393 CSMF27 44395269 IC50 = 100 nM T82393 CBG4Q5 44395271 IC50 = 1.9 nM T82393 CGKI40 44395434 IC50 = 1.6 nM T82393 C3Z6DG 44395454 IC50 = 60 nM T82393 CZB81D 44395506 IC50 = 1.6 nM T82393 CPJ4G7 44395643 IC50 = 7.1 nM T82393 CC05MG 44395660 IC50 = 73 nM T82393 CNQ6C0 44395935 IC50 = 0.48 nM T82393 C3UO7Y 44395976 IC50 = 2.5 nM T82393 CAV7Z6 44396001 IC50 = 6.5 nM T82393 CTDR73 44396048 IC50 = 3.3 nM T82393 CKV57D 44399071 IC50 = 12 nM T82393 C0NSO4 44399233 IC50 = 6.2 nM T82393 CRL5D0 44399252 IC50 = 7.3 nM T82393 CHL9S2 44399294 IC50 > 100000 nM T82393 CD49UI 44399312 IC50 > 100000 nM T82393 C7IDB0 44399341 IC50 = 5.2 nM T82393 CA0DV5 44399432 IC50 = 11 nM T82393 C95RKA 44399451 IC50 = 12 nM T82393 C3LS8N 44399509 IC50 > 100000 nM T82393 CIA8T3 44399555 IC50 = 620 nM T82393 CWL84H 44399559 IC50 = 16 nM T82393 CCIG89 44399597 IC50 = 15 nM T82393 C8YDV4 44399615 IC50 = 12 nM T82393 CV2CQ0 44399635 IC50 = 7.3 nM T82393 C5S3YZ 44399659 IC50 = 6.7 nM T82393 C7XCI6 44399665 IC50 = 10 nM T82393 CW9MD1 44399704 IC50 = 6.7 nM T82393 C2JMC1 44399712 IC50 = 17 nM T82393 CD8Q2Y 44399731 IC50 = 11 nM T82393 CC16YQ 44399733 IC50 = 10 nM T82393 C7Z0OH 44404761 IC50 = 28 nM T82393 CT7CD3 44409041 IC50 = 62 nM T82393 CJ2Q8Z 44409042 IC50 = 40 nM T82393 CY3KF2 44409047 IC50 = 53 nM T82393 CT01JW 44409066 IC50 = 74 nM T82393 CJNE37 44409163 IC50 = 153 nM T82393 CVA69I 44409164 IC50 = 199 nM T82393 C9I0JW 44409184 IC50 = 138 nM T82393 C1JSU2 44409197 IC50 = 112 nM T82393 CW4BM3 44409214 IC50 = 40 nM T82393 CVRL76 44409215 IC50 = 35 nM T82393 C9F7HR 44409221 IC50 = 42 nM T82393 CJ70LK 44409222 IC50 = 23 nM T82393 C5J1PS 44409261 IC50 = 32 nM T82393 C06EZF 44409365 IC50 = 20 nM T82393 CV5AW8 44409366 IC50 = 42 nM T82393 C9PS4Q 44409369 IC50 = 57 nM T82393 C1S4GD 44409389 IC50 = 11 nM T82393 C69CGM 44409390 IC50 = 15 nM T82393 C1SKI7 44409405 IC50 = 143 nM T82393 C5EH1T 44410935 IC50 > 3000 nM T82393 C84ZSL 44411052 Ki = 57 nM T82393 CUE29K 44411053 Ki = 321 nM T82393 C80VDP 44413972 IC50 = 2.3 nM T82393 CVM7Y3 44413975 IC50 = 2.2 nM T82393 C4X0GA 44413977 IC50 = 2 nM T82393 CH01EO 44413978 IC50 = 6 nM T82393 CQ8HK9 44413979 IC50 = 1.8 nM T82393 CBT0P2 44413982 IC50 = 2.1 nM T82393 CIJ39D 44413983 IC50 = 1.7 nM T82393 C9BA0V 44413987 IC50 = 1.4 nM T82393 CE3WP0 44413991 IC50 = 2.3 nM T82393 CDUI73 44413992 IC50 < 1 nM T82393 CH2X6W 44413997 IC50 = 2.2 nM T82393 CIL86B 44413999 IC50 = 4 nM T82393 C25XOA 44414001 IC50 = 1 nM T82393 CHN85S 44414002 IC50 = 1.4 nM T82393 C2OJ4B 44414029 IC50 = 4.9 nM T82393 CZ5KM8 44421257 IC50 = 190 nM T82393 CO24JF 44423677 IC50 = 180000 nM T82393 CK5H7O 44429877 IC50 = 12 nM T82393 CQL1X9 44429878 IC50 < 1 nM T82393 C1CYV2 44429879 IC50 = 2 nM T82393 C7AXP9 44429880 IC50 = 1.2 nM T82393 CXOS97 44429881 IC50 < 1 nM T82393 C2MQ0I 44429882 IC50 = 2.2 nM T82393 CQ5PT8 44429883 IC50 = 1.4 nM T82393 CQRO36 44429884 IC50 = 1.6 nM T82393 CM27YB 44429885 IC50 = 1.3 nM T82393 C9JH0T 44429886 IC50 = 2.8 nM T82393 CD2B3T 44429887 IC50 = 1.33 nM T82393 C6V1CO 44429888 IC50 = 5.6 nM T82393 CBC6W4 44429889 IC50 = 1.1 nM T82393 C7A0LF 44429890 IC50 < 1 nM T82393 CS0M3L 44429891 IC50 < 1 nM T82393 CX93QY 44429892 IC50 = 3 nM T82393 C7SWV1 44429893 IC50 = 7 nM T82393 C8QKS0 44429894 IC50 < 1 nM T82393 CBS47K 44429896 IC50 < 1 nM T82393 CI7TG1 44429897 IC50 = 1.8 nM T82393 CLJ48T 44429898 IC50 = 1 nM T82393 C3F9CK 44429899 IC50 = 1.2 nM T82393 C8PVF7 44429900 IC50 = 1 nM T82393 C6U0TK 44429901 IC50 = 1.5 nM T82393 CBK9M5 44429902 IC50 = 1.5 nM T82393 C72YFT 44429903 IC50 = 1.4 nM T82393 CMO9Q3 44429905 IC50 = 1.7 nM T82393 C82QFR 44431840 IC50 = 750 nM T82393 C7Q6RP 44431841 IC50 = 920 nM T82393 C0MK3W 44431842 IC50 = 96 nM T82393 CZ57SD 44431843 IC50 = 67 nM T82393 C8BHL5 44431844 IC50 = 96 nM T82393 CR1DN9 44431845 IC50 = 220 nM T82393 CHFB16 44431846 IC50 = 700 nM T82393 C0C3ZT 44431847 IC50 = 86 nM T82393 CS49GV 44431848 IC50 = 110 nM T82393 C4AVK5 44431849 IC50 = 95 nM T82393 C5DH4Q 44431850 IC50 = 120 nM T82393 CLHE45 44431851 IC50 = 50 nM T82393 CYG29L 44431852 IC50 > 3000 nM T82393 C4OF5L 44431853 IC50 = 130 nM T82393 C36SMB 44431854 IC50 = 260 nM T82393 CJZ3N6 44431855 IC50 = 78 nM T82393 CE4OI0 44431856 IC50 = 420 nM T82393 C12QOZ 44431857 IC50 = 720 nM T82393 CQ60VL 44431858 IC50 = 460 nM T82393 CBX8S0 44431859 IC50 = 230 nM T82393 CO3NE2 44431860 IC50 = 98 nM T82393 C8WBG1 44431861 IC50 = 85 nM T82393 CQ3U4H 44431862 IC50 = 1200 nM T82393 CN74TQ 44431863 IC50 = 72 nM T82393 C1S9CM 44431864 IC50 = 87 nM T82393 CY1TU8 44431865 IC50 = 77 nM T82393 CKUD90 44439848 IC50 = 0.026 nM T82393 CB9P0C 44442303 IC50 = 14 nM T82393 C7HO0Y 44442304 IC50 = 8 nM T82393 CAR3S2 44442305 IC50 = 3.2 nM T82393 CZK0A9 44442306 IC50 = 15 nM T82393 C71MCV 44442307 IC50 = 6.3 nM T82393 CN70HO 44442308 IC50 = 6 nM T82393 CVE5P0 44442309 IC50 = 5.8 nM T82393 C3PT7N 44442310 IC50 = 1.7 nM T82393 CGS18B 44442311 IC50 = 5 nM T82393 CIZL27 44442312 IC50 = 8.8 nM T82393 CCFV76 44442313 IC50 = 5.4 nM T82393 C4HYM6 44442314 IC50 = 4.1 nM T82393 CZ2PE6 44442315 IC50 = 5.9 nM T82393 C2N8BW 44442316 IC50 = 9.6 nM T82393 C3I7RG 44442317 IC50 = 62 nM T82393 CGR6E7 44442318 IC50 = 21 nM T82393 C97ZHM 44442319 IC50 = 8 nM T82393 C3DIB8 44442320 IC50 = 18 nM T82393 CP5H1Q 44446267 IC50 = 28 nM T82393 C30TQK 44446273 IC50 = 550 nM T82393 CB76CO 44446275 IC50 = 840 nM T82393 CCA8Z1 44446278 IC50 = 12400 nM T82393 CMYB26 44446280 IC50 = 36 nM T82393 C8VC3H 44446361 IC50 < 1 nM T82393 CB9W4S 44446362 Ki = 30 nM T82393 CJP64O 44446363 Ki = 17 nM T82393 CFO27Y 44478926 IC50 = 67000 nM T82393 C5D7YP 44564046 IC50 = 1 nM T82393 CIQK89 44564047 IC50 = 8 nM T82393 CR6NO2 44564180 IC50 = 28 nM T82393 CI72AB 44564406 IC50 = 25 nM T82393 C8GVR6 44564504 IC50 = 110000 nM T82393 CY1A8V 44564505 IC50 = 1 nM T82393 CWD32S 44580184 IC50 = 2.2 nM T82393 CK68GT 44580539 Ki = 61 nM T82393 C2F5ZI 44580800 Ki = 0.28 nM T82393 CXIY57 44580801 Ki = 0.36 nM T82393 C0OA8Y 44580802 Ki = 0.3 nM T82393 C5A3EG 44580803 Ki = 0.25 nM T82393 CD1VP0 44580804 Ki = 0.38 nM T82393 C41YQV 44580805 Ki = 0.54 nM T82393 CGFN68 44580806 Ki = 0.63 nM T82393 CNC4D7 44581071 Ki = 6 nM T82393 C63MNG 44581072 Ki = 5 nM T82393 C7H3SW 44581073 Ki = 158 nM T82393 CETH14 44581091 Ki = 381 nM T82393 CORS68 44581092 Ki = 3 nM T82393 C9SDP8 44581093 Ki = 2 nM T82393 CPY40M 44581094 Ki = 18 nM T82393 CDF48U 44581111 Ki = 12 nM T82393 CCT70O 44581112 Ki = 22 nM T82393 CNLK39 44581113 Ki = 37 nM T82393 CR47HS 44581138 Ki = 1 nM T82393 C1B9RT 44581139 Ki = 0.14 nM T82393 CE91OJ 44581163 Ki = 0.15 nM T82393 C1NM0F 44581164 Ki = 0.76 nM T82393 CE2XC0 44581165 Ki = 0.15 nM T82393 C84CRF 44581166 Ki = 0.21 nM T82393 CJ7IB5 44592563 IC50 = 540 nM T82393 CC6I5F 44592661 IC50 > 100000 nM T82393 CLPB12 44592662 IC50 > 100000 nM T82393 CZI95A 44592663 IC50 > 100000 nM T82393 CD4V5F 44592694 IC50 = 300 nM T82393 C6UX9Y 44592695 IC50 = 190 nM T82393 C26BCK 44592730 IC50 = 900 nM T82393 COB8I4 44592731 IC50 = 250 nM T82393 CBJL46 44592732 IC50 = 330 nM T82393 C2J0MG 44592766 IC50 = 280 nM T82393 C6X2SC 44592767 IC50 = 500 nM T82393 CN1QG3 44592768 IC50 = 490 nM T82393 C1VC8I 44592769 IC50 = 300 nM T82393 CY1IB2 44592791 IC50 = 340 nM T82393 C4WY7F 44592792 IC50 = 320 nM T82393 CJEN34 44592793 IC50 = 290 nM T82393 COR2E9 44592834 IC50 = 330 nM T82393 C48XPY 44592835 IC50 = 410 nM T82393 C0PH2U 44592836 IC50 = 470 nM T82393 CU7K0J 44592980 IC50 = 3670 nM T82393 C2B0GI 45268787 IC50 = 14000 nM T82393 CACH13 45269631 IC50 = 53000 nM T82393 C3SQL2 45378250 IC50 = 110 nM T82393 CQE49A 45378251 IC50 = 210 nM T82393 CO4AC6 45378252 IC50 = 1.6 nM T82393 C42FPG 45378253 IC50 = 0.7 nM T82393 CI82BN 45378254 IC50 = 59 nM T82393 C6MY2W 45380188 IC50 = 10000 nM T82393 C9P0DG 45380189 IC50 = 1100 nM T82393 CRY0E8 45380190 IC50 = 300 nM T82393 C0MPH3 45380191 IC50 = 44000 nM T82393 CSX5I9 46175170 IC50 = 4000 nM T82393 C56WVI 46184724 Ki = 66 nM T82393 CC1UA9 46190335 IC50 = 560 nM T82393 C9E2TX 46190374 IC50 = 281 nM T82393 CB6J4E 46190376 IC50 = 61 nM T82393 CI38EV 46190377 IC50 = 104 nM T82393 C0SF5X 46190511 IC50 = 178 nM T82393 CQ9E7N 46190515 IC50 = 92 nM T82393 CKE79Q 46190562 IC50 = 282 nM T82393 CPA19Y 46190563 IC50 = 339 nM T82393 C6KB1E 46190565 IC50 = 176 nM T82393 CEW0P1 46198901 Ki = 1.8 nM T82393 CCH49G 46198902 Ki = 0.4 nM T82393 CDBX91 46199152 Ki = 0.1 nM T82393 C9I2NM 46199503 Ki = 0.6 nM T82393 CT31MV 46200599 Ki = 0.5 nM T82393 C3ZLX1 46229743 Ki = 13 nM T82393 C5ZD8H 46229744 Ki = 33 nM T82393 CI9TC3 46229836 Ki = 93 nM T82393 C1EI5X 46229837 Ki = 70 nM T82393 CVJ5H1 46229838 Ki = 48 nM T82393 CIFE94 46229872 Ki = 8 nM T82393 C80QEZ 46229873 Ki = 461 nM T82393 CFM90S 46229874 Ki = 22 nM T82393 CA6H9C 46229924 Ki = 13 nM T82393 C10VYI 46229925 Ki = 1520 nM T82393 CF39RG 46229926 Ki = 1110 nM T82393 CK6D1T 46229976 Ki = 5530 nM T82393 CDA06S 46229977 Ki = 10600 nM T82393 C7CJA0 46230272 Ki = 1100 nM T82393 C43YOX 46230317 Ki = 1400 nM T82393 C27ECQ 46230320 Ki = 2500 nM T82393 CT2B8G 46230321 Ki = 1300 nM T82393 C6JWZ2 46230364 Ki = 1280 nM T82393 CSA85U 46230365 Ki = 1020 nM T82393 CE8XC2 46230411 Ki = 325 nM T82393 C36PZE 46230412 Ki = 20 nM T82393 CTAH67 46230413 Ki = 725 nM T82393 CY72JF 46230471 Ki = 91 nM T82393 CF7XC8 46230472 Ki = 164 nM T82393 CVAP06 46829300 Ki = 2 nM T82393 CH0Z1E 46844314 Ki = 0.4 nM T82393 CGR1Y6 46845559 Ki = 0.8 nM T82393 C7IXV6 46849757 IC50 > 10000 nM T82393 C20BTY 46856241 Ki = 0.8 nM T82393 CG7RD1 46881430 Ki = 4 nM T82393 CBX8V2 46881486 Ki = 1048 nM T82393 CK0GY2 46881487 Ki = 2729 nM T82393 C30DTL 46881488 Ki > 50000 nM T82393 C3Z6LP 46881520 Ki = 56 nM T82393 CE6S0U 46881521 Ki > 500 nM T82393 C6O0JF 46881522 Ki = 3.3 nM T82393 CHK0X4 46881523 Ki = 9 nM T82393 CS08MG 46881568 Ki = 10 nM T82393 C4TA7H 46881569 Ki = 1.6 nM T82393 C9X7OL 46881608 Ki = 0.7 nM T82393 CUJ94M 46881609 Ki = 0.7 nM T82393 C17ZEA 46881610 Ki = 1.1 nM T82393 CT6Q3B 46881611 Ki = 0.5 nM T82393 C23SXN 46881647 Ki = 2.4 nM T82393 CZHP14 46881648 Ki = 9 nM T82393 C6MDX0 46881649 Ki = 332 nM T82393 CTX73F 46881694 Ki = 1.7 nM T82393 C4VEZ3 46882679 IC50 = 2700 nM T82393 C0S9WB 46919610 Ki = 4 nM T82393 COI75X 46933693 Ki = 0.2 nM T82393 CZD97B 46933694 Ki = 0.5 nM T82393 C9SRJ4 46933999 Ki = 0.1 nM T82393 C6IVW3 46934000 Ki = 0.77 nM T82393 CD15NF 49854511 IC50 = 210 nM T82393 C1Y6CT 49864868 Ki = 3 nM T82393 C1EXH5 49864904 Ki = 7 nM T82393 CV82ZG 49864905 Ki = 8 nM T82393 CI3UX1 49864906 Ki = 6 nM T82393 C49XVF 49864939 Ki = 6 nM T82393 CQI43E 49864940 Ki = 29 nM T82393 C0D4BO 49864941 Ki = 27 nM T82393 C49ZNY 49864990 Ki = 2 nM T82393 C79NYS 49864991 Ki = 18 nM T82393 CA6RD8 49864992 Ki = 9 nM T82393 C3DW8Z 49864993 Ki = 3 nM T82393 CC28UG 49865044 Ki = 0.5 nM T82393 CGA4S3 49865045 Ki = 0.6 nM T82393 CM43AH 49865046 Ki = 1.4 nM T82393 CI5X9A 49865107 Ki = 0.9 nM T82393 CT0D7O 49865108 Ki = 0.6 nM T82393 CYD0Z3 49865165 Ki = 1.2 nM T82393 C83RDH 49865166 Ki = 1 nM T82393 C05BHN 49865167 Ki = 0.5 nM T82393 CLUT34 49865168 Ki = 0.88 nM T82393 CR82AJ 49865223 Ki = 2.6 nM T82393 C4Q1NC 49865224 Ki = 2 nM T82393 C6SPT2 49865225 Ki = 3 nM T82393 CQI4T3 49865286 Ki = 0.8 nM T82393 C3CAP0 49865287 Ki = 2 nM T82393 CI89DJ 49865288 Ki = 31 nM T82393 C7UO5N 49865338 Ki = 28 nM T82393 CH69DC 49865339 Ki = 10 nM T82393 CUD7O0 50941549 IC50 > 10000 nM T82393 CXF4V3 50990921 IC50 = 250 nM T82393 C51GVO 51035425 Ki = 0.4 nM T82393 CU2SX3 51355576 Ki > 10000 nM T82393 CPGA06 52941225 Ki = 0.92 nM T82393 CXR8E7 52941250 Ki = 0.07 nM T82393 CR60IV 52941256 Ki = 0.5 nM T82393 COTL14 52941292 Ki = 2.78 nM T82393 CFX27S 52941303 Ki = 0.17 nM T82393 C2SFK1 52942472 Ki = 0.22 nM T82393 CC38VH 52942483 Ki = 0.13 nM T82393 CN0I6V 52942509 Ki = 0.56 nM T82393 C2W6UV 52942531 Ki = 0.19 nM T82393 C25JRD 52943632 Ki = 0.16 nM T82393 C73HML 52943705 Ki = 2.55 nM T82393 C09NZH 52944849 Ki = 0.47 nM T82393 CFT09H 52944923 Ki = 0.5 nM T82393 CF8O1M 52945321 Ki = 0.53 nM T82393 C17FYL 52946125 Ki = 2 nM T82393 CI15CF 52947303 Ki = 0.29 nM T82393 C0MNC8 52947338 Ki = 0.41 nM T82393 C81HAL 52947372 Ki = 0.85 nM T82393 CBO75P 52947420 Ki = 0.6 nM T82393 CPLD94 52948549 Ki = 0.14 nM T82393 CEJ90S 52949743 Ki = 0.61 nM T82393 C0XTZ3 52949779 Ki = 0.72 nM T82393 C3J5RK 52949816 Ki = 0.42 nM T82393 CMV85W 52950115 Ki = 2.35 nM T82393 C1Y5UN 52951473 IC50 > 10000 nM T82393 C8J9EM 52951589 IC50 > 10000 nM T82393 CEAS70 52951591 IC50 > 10000 nM T82393 C4DG1F 52951593 IC50 > 10000 nM T82393 C6XJ3V 52951596 IC50 > 10000 nM T82393 C9U3AF 52951710 IC50 > 10000 nM T82393 C4M1CA 52951712 IC50 > 10000 nM T82393 C76LDY 52951967 IC50 = 1600 nM T82393 CYKS94 52951968 IC50 > 10000 nM T82393 CE0FP3 52951969 IC50 > 10000 nM T82393 CL69OM 52951970 IC50 > 10000 nM T82393 CMPB74 52951971 IC50 = 3800 nM T82393 CZ1TN8 52951972 IC50 = 1100 nM T82393 CK08OB 52952074 IC50 = 1900 nM T82393 C46AYR 52952075 IC50 > 10000 nM T82393 CR32ZW 52952076 IC50 > 10000 nM T82393 CJ9O3S 52952077 IC50 > 10000 nM T82393 C3N9TF 52952078 IC50 > 10000 nM T82393 CE4Q7F 52952273 IC50 > 10000 nM T82393 CMA69V 52952274 IC50 > 10000 nM T82393 C7KB5W 52952275 IC50 > 10000 nM T82393 CRO0X4 52952276 IC50 > 10000 nM T82393 CSJ05E 52952277 IC50 > 10000 nM T82393 C29UJB 52952388 IC50 > 10000 nM T82393 C3H5ID 52952389 IC50 > 10000 nM T82393 CSX69R 52952390 IC50 > 10000 nM T82393 CB36KP 52952492 IC50 > 10000 nM T82393 C67OEU 52952493 IC50 = 6300 nM T82393 CV1I0A 52952597 IC50 > 10000 nM T82393 CGI87K 52952598 IC50 > 10000 nM T82393 CXWI18 52952599 IC50 > 10000 nM T82393 C46VHP 52952600 IC50 > 10000 nM T82393 CH3G6R 52952601 IC50 > 10000 nM T82393 CC0Y3M 52952602 IC50 > 10000 nM T82393 C2T9DN 53232907 Ki = 7 nM T82393 C2HG9L 53232908 Ki = 7 nM T82393 CU13LN 53233013 Ki = 4 nM T82393 C5VR6F 53233014 Ki = 17 nM T82393 C3BGW0 53233015 Ki = 5 nM T82393 C4G5QR 53233016 Ki = 4 nM T82393 CS76AR 53233128 Ki = 0.5 nM T82393 CN0VD1 53316692 IC50 = 0.9 nM T82393 C47DIU 53318911 IC50 = 21 nM T82393 CC6DR2 53318912 IC50 = 22 nM T82393 C7V1NC 53320225 IC50 = 420 nM T82393 CVH2B7 53320226 IC50 = 27000 nM T82393 CO8QK2 53320227 IC50 = 5500 nM T82393 C5HYA4 53320636 IC50 = 0.46 nM T82393 CTQ02K 53320639 IC50 = 12 nM T82393 CNS3F2 53321542 IC50 = 19 nM T82393 CSYW40 53322877 IC50 = 1400 nM T82393 C3QHA6 53322879 IC50 = 3000 nM T82393 C0H7FQ 53324260 IC50 = 2800 nM T82393 C4G1HK 53325498 IC50 = 3200 nM T82393 CO5L1I 53325499 IC50 = 230 nM T82393 CM53CG 53326761 IC50 = 24000 nM T82393 C6Y2EV 53374826 IC50 = 21500 nM T82393 CBL30Y 54181369 IC50 = 17 nM T82393 CQN6W7 54580563 Ki = 8 nM T82393 CE8JM6 54580564 Ki = 9 nM T82393 CK25TE 54580565 Ki = 0.2 nM T82393 CK3WC6 54580566 Ki = 307 nM T82393 CGMH73 54581562 Ki = 6 nM T82393 C6VB8S 54581563 Ki = 36 nM T82393 CQPI21 54581564 Ki = 15 nM T82393 C5CN9T 54581565 Ki = 5 nM T82393 CUVG19 54581885 Ki = 0.9 nM T82393 C6PD2K 54581886 Ki = 2 nM T82393 C0AX7O 54581923 Ki = 6 nM T82393 CJ57VO 54581924 Ki = 4 nM T82393 CKD41A 54582559 Ki = 37 nM T82393 CQ9M4H 54582560 Ki = 37 nM T82393 CXQ9B3 54582561 Ki = 36 nM T82393 C0ZXQ3 54582562 Ki = 2 nM T82393 CY2VT0 54582563 Ki = 315 nM T82393 C2D4CL 54582564 Ki = 2 nM T82393 CS8V9X 54582565 Ki = 74 nM T82393 CN63KE 54582810 Ki = 0.5 nM T82393 CO46BU 54582811 Ki = 14 nM T82393 CM9QB0 54582812 Ki = 65 nM T82393 C7KDS5 54582833 Ki = 1 nM T82393 C97ZWN 54582834 Ki = 2 nM T82393 C9SHY2 54582835 Ki = 0.6 nM T82393 C2BUK8 54582836 Ki = 1 nM T82393 CIN9R0 54583526 Ki = 9.3 nM T82393 C9U3TE 54583527 Ki = 2 nM T82393 CO9GD2 54583528 Ki = 12 nM T82393 CX1HD2 54583529 Ki = 13 nM T82393 COI4W7 54583579 Ki = 3 nM T82393 CLQ2F5 54583813 Ki = 6.7 nM T82393 CJ8P7H 54583814 Ki = 38 nM T82393 CA48DY 54583815 Ki = 4 nM T82393 C83EFJ 54583816 Ki = 10 nM T82393 CNW23D 54583850 Ki = 9 nM T82393 C5Z3UG 54584508 Ki = 17 nM T82393 CWL2Q1 54584509 Ki = 28 nM T82393 CP7QN3 54584510 Ki = 8 nM T82393 CK26IR 54584511 Ki = 296 nM T82393 CX69PA 54584787 Ki = 7.6 nM T82393 CS9GC0 54584788 Ki = 5 nM T82393 C18SHQ 54584805 Ki = 531 nM T82393 C53ERM 54585452 Ki = 48 nM T82393 C45ISX 54585453 Ki = 12 nM T82393 C8DWZ4 54585754 Ki = 16 nM T82393 C69DUF 54586417 Ki = 3 nM T82393 CS8B2I 54586418 Ki = 11 nM T82393 C6PB9M 54586419 Ki = 4 nM T82393 C7IE5K 54586420 Ki = 4 nM T82393 CTW20Y 54586421 Ki = 22 nM T82393 C31BJF 54586422 Ki = 4 nM T82393 CML08P 54586423 Ki = 270 nM T82393 CZ5M0H 54586703 Ki = 0.4 nM T82393 CU7B1L 54586704 Ki = 10 nM T82393 C4L0FV 54586705 Ki = 6 nM T82393 C2RIK0 54586706 Ki = 39 nM T82393 CL9UJ3 54586736 Ki = 2 nM T82393 CA8U9G 54586737 Ki = 2 nM T82393 CL08RB 54586738 Ki = 2 nM T82393 CZ5WQ7 54587440 Ki = 20 nM T82393 CB2Y3Q 54587441 Ki = 0.5 nM T82393 CK4B0E 54587442 Ki = 18 nM T82393 CD5LK7 54587443 Ki = 45 nM T82393 C87WOJ 54587742 Ki = 87 nM T82393 C28RBQ 54587743 Ki = 22 nM T82393 C3I6FW 54587744 Ki = 2.6 nM T82393 CEZ5C6 54587745 Ki = 1 nM T82393 CL9SC3 54587769 Ki = 1 nM T82393 CGH0S7 54589400 IC50 > 100000 nM T82393 CN39JQ 56661881 IC50 = 280 nM T82393 C8O0VH 56665352 IC50 = 80 nM T82393 C5BC4N 56678961 IC50 = 160 nM T82393 C41RYI 56678962 IC50 = 126 nM T82393 C5MNW4 56678963 IC50 = 70 nM T82393 C2CJ3I 56678964 IC50 = 74 nM T82393 CKJ9S1 56835167 IC50 = 10000 nM T82393 C21CLZ 56835168 IC50 = 16000 nM T82393 C0L2TS 56835169 IC50 = 33000 nM T82393 C10BMZ 57127110 IC50 = 48 nM T82393 CHJ78V 57561223 Ki = 1.4 nM T82393 CS9D6I 57561259 Ki = 0.5 nM T82393 CXU65J 57561279 Ki = 0.5 nM T82393 CWH7V8 57561293 Ki = 0.7 nM T82393 CSO90P 57561300 Ki = 2 nM T82393 CA7P3O 57561339 Ki = 1.6 nM T82393 CFGD84 57561367 Ki = 0.7 nM T82393 CW68ZR 57561449 Ki = 3.6 nM T82393 CY1N3J 57792153 IC50 = 2.1 nM T82393 C5RK1A 57848896 IC50 = 199.53 nM T82393 C50SEX 57848902 IC50 = 0.1 nM T82393 C48MLO 57848904 IC50 = 2.4 nM T82393 C3QX4R 57848908 IC50 = 3.7 nM T82393 CFUB46 57848909 IC50 = 19 nM T82393 CMU19B 57848917 IC50 = 6.31 nM T82393 COT20V 57848922 IC50 = 1 nM T82393 CS5OJ1 57848924 IC50 = 0.6 nM T82393 CTH56Z 57848925 IC50 = 1 nM T82393 C9GZ0L 58053137 Ki = 0.4 nM T82393 CM43LS 58053165 Ki = 0.9 nM T82393 CE8Q7X 58053190 Ki = 0.5 nM T82393 C18GIT 58053321 Ki = 1.3 nM T82393 CM98QB 58053362 Ki = 0.4 nM T82393 C7WPS1 58053551 Ki = 2.5 nM T82393 CT72DF 58053577 Ki = 1.9 nM T82393 CP4UO7 58053649 Ki = 0.2 nM T82393 C5CJ6D 58053678 Ki = 0.2 nM T82393 CR9LZ8 58053823 Ki = 0.5 nM T82393 C2KT6W 58054076 Ki = 0.3 nM T82393 C2EPW3 58521428 IC50 = 156 nM T82393 C0I9GJ 58521444 IC50 = 141 nM T82393 CRO3Q0 58521447 IC50 = 7150 nM T82393 C52ESR 66559934 IC50 > 50000 nM T82393 C57ARI 66560021 IC50 > 50000 nM T82393 CU58DB 66560022 IC50 > 50000 nM T82393 C16RDM 66560389 IC50 = 12600 nM T82393 C8RZG9 66560479 IC50 = 19900 nM T82393 CS5J6B 68081093 Ki = 0.4 nM T82393 C0S1ZQ 70232814 Ki = 0.4 nM T82393 CA17KW 70234871 Ki = 0.4 nM T82393 CQV08A 70235355 Ki = 0.7 nM T82393 C17UGK 70235517 Ki = 1 nM T82393 C59NWG 70236065 Ki = 0.5 nM T82393 CKW2Q5 71453375 IC50 = 7900 nM T82393 C7RZN9 71652216 IC50 = 590 nM T82393 C7YFC8 72711513 IC50 = 500 nM T82393 CTM4P2 72713638 IC50 = 16 nM T82393 C0N2JX 72713639 IC50 = 145 nM T82393 CF4K8Y 72713862 IC50 = 200 nM T82393 C3R6JO 72713863 IC50 = 640 nM T82393 CW9D3V 72713864 IC50 = 104 nM T82393 CQ6FH3 72713865 IC50 = 71 nM T82393 C4FYB0 72713866 IC50 = 280 nM T82393 CH6SI1 72713867 IC50 = 76 nM T82393 CS21QM 72713868 IC50 = 650 nM T82393 CB56AP 72714081 IC50 = 82 nM T82393 C1CK0E 72714082 IC50 = 840 nM T82393 CP5Q8W 72714083 IC50 = 160 nM T82393 CA03NU 72714084 IC50 > 50000 nM T82393 CRUH64 72714085 IC50 = 320 nM T82393 CZFY06 72714322 IC50 = 43 nM T82393 CDY70J 72714323 IC50 = 11 nM T82393 CD56BA 72714324 IC50 = 1.9 nM T82393 CW01EA 73349535 IC50 > 10000 nM T82393 C21FEO 76331549 IC50 = 669 nM T82393 CX39OW 76331563 IC50 = 48 nM T82393 C9CY5K 76335167 IC50 = 764 nM T82393 C5LB0U 78426619 IC50 = 5400 nM T82393 CET6N8 78426757 IC50 = 11000 nM T82393 CGQ8F3 86287515 IC50 = 10000 nM T82393 CJ37XE 86287516 IC50 = 10000 nM T82393 COV8I9 86291010 IC50 = 2.3 nM T82393 C3EIU0 86607902 IC50 = 0.6 nM T82393 CAB2F5 87349434 Ki = 900 nM T82393 C80HRG 87586471 IC50 = 0.6 nM T82393 CUK9O0 87586520 IC50 = 1.8 nM T82393 C7K9UA 87586626 IC50 = 0.631 nM T82393 CEN92C 87587735 IC50 = 61 nM T82393 C3O8UP 88272565 IC50 = 1 nM T82393 CRT54C 101910871 IC50 = 10000 nM T82393 C1J3CK 117094707 IC50 = 1500 nM T82393 C1W5NH 118718816 IC50 = 12 nM T82393 C5ZS4E 118722686 IC50 = 5400 nM T82393 CGY9V6 122181846 IC50 = 10000 nM T82393 C3GOS2 122181847 IC50 = 10000 nM T82393 CN7WC6 122181848 IC50 = 29000 nM T82393 CJ7B4Y 122181849 IC50 = 94000 nM T82393 CJNH05 122181850 IC50 = 15000 nM T82393 C2KU3W 122181851 IC50 = 5900 nM T82393 CO6N5R 122181852 IC50 = 35000 nM T82393 CN7XR8 122181988 IC50 = 5400 nM T82393 C8DHI1 122181989 IC50 = 10000 nM T82393 C9XDO5 122181990 IC50 = 7900 nM T82393 CP4M8S 122181991 IC50 = 6500 nM T82393 CT8XW5 122181992 IC50 = 8100 nM T82393 C06QZX 122181993 IC50 = 15000 nM T82393 C9G0QI 122181994 IC50 = 8400 nM T82393 C9RVB8 122181995 IC50 = 5700 nM T82393 CLCW15 122181996 IC50 = 5700 nM T82393 CT7D4F 122181997 IC50 = 1900 nM T82393 CZO32N 122181998 IC50 = 4300 nM T82393 C40DWG 122181999 IC50 = 8500 nM T82393 CT03QA 127026888 IC50 = 90 nM T82393 CWI7K3 127037444 IC50 = 150000 nM T82393 C9QLI2 127037445 IC50 = 9500 nM T82393 CCA0R8 127037446 IC50 = 114000 nM T82393 C8R6UN 130273543 IC50 = 8 nM T82393 C29FSJ 130273545 IC50 = 61 nM T82393 CJC92A 130273554 IC50 = 4.6 nM T82393 C3FZ8V 130273583 IC50 = 33 nM T82393 CSY1E4 130273592 IC50 = 6 nM T82393 CGU7I0 130273655 IC50 = 16 nM T82393 CPE48N 130275134 IC50 = 6 nM T82393 CBF3E1 130275145 IC50 = 5 nM T82393 CSR3Q6 130282545 IC50 = 790 nM T82393 C8JS5P 130282613 IC50 = 37 nM T82393 C1S2NX 130282614 IC50 = 590 nM T82393 CYA92R 130282633 IC50 = 4 nM T82393 CO3QE2 130282636 IC50 = 20 nM T82393 C2HF7Z 130282889 IC50 = 31 nM T82393 CTN42D 132941363 IC50 = 10000 nM T82393 CHV2U1 135438561 IC50 > 10000 nM T82393 CRAZ20 135485671 IC50 = 0.57 nM T82393 C2URS4 135501193 IC50 = 12 nM T82393 CY3DQ8 135506889 IC50 = 3.4 nM T82393 CF5V0O 135518749 IC50 = 2400 nM T82393 CRA5P8 135518776 IC50 = 0.33 nM T82393 CT23GK 136032622 Ki = 0.18 nM T82393 CA5JR6 136054481 IC50 > 10000 nM T82393 CV47JN 136054485 IC50 > 10000 nM T82393 CZ48WO 136054487 IC50 > 10000 nM T82393 C8FGT0 136054495 IC50 > 10000 nM T82393 CG70BZ 136054516 IC50 > 10000 nM T82393 CSM57W 136054520 IC50 = 510 nM T82393 C4MIH8 136059691 IC50 = 4.3 nM T82393 CXNG40 136118011 IC50 = 439 nM T82393 C1IOH9 136118012 IC50 = 34 nM T82393 CTY79S 136118013 IC50 > 1000 nM T82393 CTE87J 136118014 IC50 = 162 nM T82393 CJG54U 136219136 IC50 = 16000 nM T82393 C3CAV5 136219141 IC50 > 30000 nM T82393 CPB07Z 136241630 IC50 = 21000 nM T82393 CIEW62 136380958 IC50 > 10000 nM T82393 C9HS7J 137287436 IC50 > 10000 nM T82393 C3QZ8E 137631527 IC50 = 60 nM T82393 CHN37C 137631926 IC50 = 35 nM T82393 C5U9TO 137631966 IC50 = 26 nM T82393 C0D1HT 137632332 IC50 = 3600 nM T82393 CMZ2U5 137632423 Ki = 0.4 nM T82393 CW20RK 137633040 IC50 = 870 nM T82393 CN95XB 137633310 IC50 = 1000 nM T82393 COA8T6 137633887 IC50 = 13 nM T82393 CMK50Q 137634170 IC50 = 71 nM T82393 CL90EH 137634282 IC50 = 6 nM T82393 CEKU45 137634768 IC50 = 150 nM T82393 CAR1Z5 137635202 IC50 = 35 nM T82393 C1I2HL 137635814 IC50 = 3.8 nM T82393 CX6O5H 137636272 IC50 = 29 nM T82393 CV82XA 137636843 IC50 = 940 nM T82393 C8KLI6 137637522 IC50 = 1200 nM T82393 C35JNR 137637606 IC50 = 9500 nM T82393 C0YHM6 137637675 IC50 = 794.33 nM T82393 CWQH36 137637804 IC50 = 6200 nM T82393 CN3P2T 137638567 IC50 = 316.23 nM T82393 CY78SL 137638706 IC50 = 23 nM T82393 CPN0H7 137639172 IC50 = 200 nM T82393 CAN0B2 137639286 IC50 = 160 nM T82393 C7TJ4H 137639420 IC50 > 10000 nM T82393 CA20NW 137639584 IC50 = 42 nM T82393 CH2UO7 137641291 IC50 = 39.81 nM T82393 C3K1CH 137641350 Ki = 1200 nM T82393 C1F3KO 137641743 IC50 > 10000 nM T82393 CI89NB 137641769 IC50 = 501.19 nM T82393 CXH06N 137641838 IC50 = 180 nM T82393 CF98BN 137642614 IC50 = 770 nM T82393 C7S3NE 137643530 IC50 = 7200 nM T82393 CE7RC6 137643560 IC50 = 24500 nM T82393 C60KGV 137643749 IC50 = 30 nM T82393 CX0PE5 137643973 IC50 = 10000 nM T82393 CO2FB5 137645222 IC50 = 1900 nM T82393 C24VDT 137645542 IC50 = 16 nM T82393 C9SLP2 137645623 IC50 = 16 nM T82393 C2TB0M 137645962 IC50 = 750 nM T82393 CM6F0N 137646068 IC50 = 5011.87 nM T82393 COX50I 137648094 IC50 > 10000 nM T82393 CD87RG 137648616 IC50 = 900 nM T82393 C5JH1B 137649848 IC50 = 350 nM T82393 C61MRQ 137650294 IC50 = 3857 nM T82393 CH2K1D 137650845 IC50 = 2900 nM T82393 C9CIY6 137651719 IC50 = 1240 nM T82393 C7YS3Z 137652101 IC50 = 210 nM T82393 C2QD3H 137652156 IC50 = 1500 nM T82393 CVP4J7 137652819 IC50 = 84 nM T82393 CRO5K4 137652849 IC50 = 7943.28 nM T82393 C6Z4EW 137653004 IC50 = 760 nM T82393 C8WS4L 137653115 IC50 = 23 nM T82393 C4T7NL 137653444 IC50 = 40 nM T82393 CF3CA4 137653882 IC50 > 10000 nM T82393 CP4SJ8 137654048 IC50 = 1145 nM T82393 CP7X4V 137654254 IC50 = 19 nM T82393 CY5EZ4 137654626 IC50 = 1197 nM T82393 C02QKF 137655494 IC50 = 14 nM T82393 C7W4VJ 137657340 IC50 = 6500 nM T82393 CBQY48 137657825 IC50 = 0.6 nM T82393 CG7ED9 137657827 IC50 > 10000 nM T82393 CI85DX 137658315 IC50 = 950 nM T82393 C7OK2V 137658353 IC50 = 1127 nM T82393 C28LGI 137658795 IC50 = 3981.07 nM T82393 C2MG8Y 137659221 IC50 > 10000 nM T82393 CUEZ46 137659996 IC50 > 10000 nM T82393 C3OE2G 137660105 IC50 = 4500 nM T82393 C4JMQ9 137660408 IC50 = 40 nM T82393 CAB7Q6 137660566 IC50 = 12 nM T82393 CS9FT7 137661162 IC50 = 672 nM T82393 CF7J6V 137662109 IC50 = 110 nM T82393 C1IUV8 145964890 IC50 = 100 nM T82393 C2VO3P 145965182 IC50 = 84 nM T82393 C1Y5WV 145965955 IC50 = 68 nM T82393 CTOV93 145966382 IC50 = 240 nM T82393 C6MUV3 145966657 IC50 = 36 nM T82393 CC6XV9 145966850 IC50 > 10000 nM T82393 CVH0L8 145967193 IC50 = 10 nM T82393 CA3B6Q 145967216 IC50 = 13 nM T82393 CGO4Z2 145967532 IC50 = 27 nM T82393 CQI8S0 145968704 IC50 = 30 nM T82393 CCI7T1 145969141 IC50 = 720 nM T82393 C65OFP 145971429 IC50 = 12 nM T82393 CN6L0Z 145971797 IC50 = 82 nM T82393 CF37VH 145972747 IC50 > 10000 nM T82393 CPZ6C2 145973916 IC50 = 210 nM T82393 CBO41G 145974267 IC50 = 1300 nM T82393 CN3G8U 145975584 IC50 = 43 nM T82393 C62ZLM 145975639 IC50 = 2300 nM T82393 C1CW5E 145976264 IC50 = 42 nM T82393 CTB0K3 145977602 IC50 = 140 nM T82393 CGD14L 145977705 IC50 = 10 nM T82393 C91ASZ 145977730 IC50 = 4 nM T82393 CF8WV2 155511139 IC50 = 541 nM T82393 CZ25LW 155512044 IC50 = 10000 nM T82393 CP9YX2 155567218 IC50 = 8900 nM T82393 C8D5VK 155567855 IC50 = 10000 nM T82393 CUL0X5 87587813 IC50 = 1.259 nM T82393 D00RNA 44446270 IC50 = 150 nM T82393 D02UYR 9907830 Ki = 3.8 nM T82393 D03AMR 9849669 Ki = 4 nM T82393 D03WJG 9910222 Ki = 2.3 nM T82393 D04WWO 9889867 IC50 = 6.2 nM T82393 D06EHW 11625778 IC50 = 14 nM T82393 D07GEL 10344307 IC50 = 220 nM T82393 D08ICI 44446277 IC50 = 110 nM T82393 D09GLA 4368 IC50 = 231 nM T82393 D09ZOA 25049753 IC50 = 2400 nM T82393 D0A4TC 446504 IC50 = 160 nM T82393 D0B3UN 44580458 Ki > 100000 nM T82393 D0G3YZ 11391583 IC50 > 98000 nM T82393 D0H2PA 9886977 Ki = 0.6 nM T82393 D0H6CK 10160968 IC50 = 36 nM T82393 D0NV9C 22004198 IC50 = 3900 nM T82393 D0Q4TA 10044321 IC50 > 100000 nM T82393 D0T1FR 44457233 IC50 > 100000 nM T82393 D0W2UK 6914621 Ki = 0.06 nM T82393 D0XK7G 10445302 IC50 = 1800 nM T82393 D0Y1XM 44423686 IC50 = 100000 nM T82393 D0Y5IQ 44255320 IC50 = 1230 nM T03917 D01XNB 4594 IC50 = 31622.78 nM T03917 D02OZE 2724385 IC50 = 400 nM T03917 D0AR3J 439501 IC50 = 3.4 ug.mL-1 T03917 D0M3QP 441207 IC50 = 8 nM T03917 D0T6XX 4679 IC50 = 199526.23 nM T03917 D08UUK 153976 IC50 = 1500 nM T03917 C2KJI7 3883 IC50 = 39810.72 nM T03917 C8A5QG 126974 IC50 = 39810.72 nM T03917 CS1W8P 126981 IC50 = 25118.86 nM T03917 C8SO6R 513481 IC50 > 150000 nM T03917 CVF85S 9885247 IC50 = 2500 nM T03917 CB1AC5 9886003 IC50 = 100 nM T03917 CGK31E 9976847 IC50 = 1000 nM T03917 C4T0QC 9987588 Ki = 320 nM T03917 CB45YI 9993694 IC50 > 150000 nM T03917 CXFO23 10042024 IC50 = 800 nM T03917 C90TJL 10056772 IC50 > 100000 nM T03917 CTA21F 10064069 IC50 = 1300 nM T03917 CWR72T 10066501 IC50 = 1600 nM T03917 C6YPS2 10069116 IC50 = 40 nM T03917 CTD8M6 10102761 IC50 > 100000 nM T03917 CM65TE 10245895 IC50 = 2100 nM T03917 CA90VD 10315757 IC50 = 1000 nM T03917 C0MG9R 10418023 IC50 > 100000 nM T03917 CG1YK0 10441258 IC50 > 100000 nM T03917 C5SKI6 10470916 IC50 = 3.6 ug.mL-1 T03917 C5TE1B 10500563 IC50 = 10000 nM T03917 CM64BU 10502985 IC50 = 31622.78 nM T03917 CA90KQ 10526174 IC50 > 100000 nM T03917 CSI28D 10548622 IC50 = 19952.62 nM T03917 CE5HY0 10549844 IC50 = 19952.62 nM T03917 C7B9YL 10595652 IC50 = 4000 nM T03917 CX60CL 10596400 IC50 = 80 nM T03917 CB2A9W 10597390 IC50 = 16 nM T03917 CTNS40 10647308 IC50 = 6309.57 nM T03917 CK1JC0 10665493 IC50 = 32000 nM T03917 C57KNH 10669035 IC50 = 6300 nM T03917 C1U3BV 10669094 IC50 = 40 nM T03917 C3I8JW 10669386 IC50 = 25118.86 nM T03917 C8SAZ1 10670402 IC50 = 25 nM T03917 CG6ZX8 10670404 IC50 = 160000 nM T03917 CB76PQ 10693245 IC50 = 251.19 nM T03917 CKC05Y 10716167 IC50 = 10000 nM T03917 CKP0Z6 10716333 IC50 > 100000 nM T03917 CSIT17 10739286 IC50 > 100000 nM T03917 CV7IG9 10739352 IC50 > 100000 nM T03917 CTLN73 10740180 IC50 = 1995.26 nM T03917 CA0D9V 10740703 IC50 > 10000 nM T03917 CD0A1E 10740783 IC50 = 7900 nM T03917 CAL1B7 10761299 IC50 > 100000 nM T03917 C62PEG 10763980 IC50 = 1000 nM T03917 C87FSR 10764407 IC50 = 1000 nM T03917 CJ2D5Z 10786633 IC50 = 199.53 nM T03917 C7KM3D 10787794 IC50 = 1995.26 nM T03917 CJ2QZ3 10834968 IC50 = 199.53 nM T03917 CO37JG 10835932 IC50 = 630 nM T03917 CN7QB9 10836552 IC50 = 6300 nM T03917 C5GT7D 10860933 IC50 = 16000 nM T03917 CUHK27 10874510 IC50 = 2000 nM T03917 CDE12N 10884700 IC50 = 3200 nM T03917 CQR9P5 10894086 IC50 = 5000 nM T03917 COQ4P3 10895365 IC50 = 3200 nM T03917 CP26SQ 10904400 IC50 = 50000 nM T03917 CZU9F6 10904597 IC50 = 100000 nM T03917 C7AE1L 10914952 IC50 = 13000 nM T03917 C67KFV 10925984 IC50 > 100000 nM T03917 CR2L9B 10926178 IC50 > 100000 nM T03917 CNSD51 10926441 IC50 = 5000 nM T03917 CB54IS 10927644 IC50 = 1000 nM T03917 C7YVU1 10938704 IC50 = 6300 nM T03917 CJT38O 10939357 IC50 = 1300 nM T03917 C4Y6CD 10949677 IC50 = 1000 nM T03917 CO5IB1 10949850 IC50 = 250 nM T03917 CC2K0R 10958069 IC50 = 4000 nM T03917 C4D8ZN 10961051 IC50 > 100000 nM T03917 CBR76K 10970799 IC50 = 8000 nM T03917 C93JRQ 10972073 IC50 = 1000 nM T03917 CM0L7R 10980156 IC50 = 63000 nM T03917 C56GKL 10991584 IC50 = 2500 nM T03917 CHEQ56 11015311 IC50 = 3200 nM T03917 CDE5F4 11027049 IC50 = 5000 nM T03917 CEXB84 11036723 IC50 > 100000 nM T03917 CAZ81O 11067985 IC50 = 2500 nM T03917 COG29B 11068897 IC50 = 10000 nM T03917 C5BIM9 11069563 IC50 = 20000 nM T03917 CCJ8A5 11070164 IC50 = 10000 nM T03917 C8E7PR 11080614 IC50 = 2500 nM T03917 CFO89W 11080939 IC50 = 3200 nM T03917 CBS0V9 11090473 IC50 = 400 nM T03917 C8FOC1 11101584 IC50 = 1600 nM T03917 CZT9U8 11112293 IC50 = 200 nM T03917 CDG8J6 11121963 IC50 = 10000 nM T03917 C21SMR 11122663 IC50 = 800 nM T03917 C24KHY 11269080 IC50 > 316227.77 nM T03917 CQS3D5 11549949 IC50 > 100 ug.mL-1 T03917 CP9Q1T 11658230 IC50 > 100 ug.mL-1 T03917 C8ZE3D 11728228 IC50 = 4000 nM T03917 C19STK 11729892 IC50 = 13000 nM T03917 CA0Y4K 11744503 IC50 = 44000 nM T03917 CCFZ87 11759494 IC50 = 800 nM T03917 CWI27U 11760135 IC50 = 3200 nM T03917 C2NHL7 11760136 IC50 = 10000 nM T03917 CDMT64 11760644 IC50 = 400 nM T03917 CFM15H 11783235 IC50 = 8000 nM T03917 CBV86W 11784165 IC50 = 50 nM T03917 CK01CJ 11812392 IC50 > 100000 nM T03917 C36CGT 11961867 IC50 = 7.04 nM T03917 C5NSE7 12038807 IC50 = 99000 nM T03917 CHW42J 12038808 IC50 = 88000 nM T03917 C1D5MK 12308635 IC50 = 4.79 nM T03917 CK60WT 12313935 IC50 = 1090 nM T03917 CZ4EF3 14019702 IC50 = 60 ug.mL-1 T03917 C5BHA7 14019705 IC50 > 100 ug.mL-1 T03917 CT1P2Z 15163488 IC50 = 25118.86 nM T03917 CPS67D 15163489 IC50 = 50118.72 nM T03917 CT2O8F 15163490 IC50 = 39810.72 nM T03917 CO6B1Y 15163491 IC50 = 6309.57 nM T03917 CZY0X9 15163492 IC50 = 316227.77 nM T03917 C3KXD9 15163493 IC50 = 50118.72 nM T03917 CN90GC 15163494 IC50 = 3981.07 nM T03917 C18YHB 15163495 IC50 = 158489.32 nM T03917 CPF38Y 15163496 IC50 > 1000000 nM T03917 CC9L8W 15163497 IC50 = 63095.73 nM T03917 CQS19H 15163498 IC50 = 3162.28 nM T03917 C38WMN 15163499 IC50 = 3162.28 nM T03917 CCHZ08 15163500 IC50 = 251188.64 nM T03917 CMLY48 15163501 IC50 > 1000000 nM T03917 CH80ZD 15163502 IC50 = 251188.64 nM T03917 CH8I3Q 15163503 IC50 = 10000 nM T03917 CZ9D1S 15163504 IC50 = 398107.17 nM T03917 CGHI34 15163505 IC50 = 19952.62 nM T03917 CMD60R 15163510 IC50 > 1000000 nM T03917 CPC2B7 15163511 IC50 > 1000000 nM T03917 C9KI7L 15406360 IC50 > 10000 nM T03917 CK2H4B 18184703 IC50 = 10000 nM T03917 CCG8T9 21576266 IC50 > 100000 nM T03917 CXW5E4 21606558 IC50 > 100 ug.mL-1 T03917 CK4ZI1 21606559 IC50 > 100 ug.mL-1 T03917 CI4C6Z 23254267 IC50 > 100000 nM T03917 CTJ0R1 23426012 IC50 = 5000 nM T03917 CXY47R 23716625 IC50 = 5000 nM T03917 CGJ2L8 44236689 IC50 > 100000 nM T03917 CEVW34 44285553 IC50 = 33000 nM T03917 C0NTH5 44285568 IC50 = 14000 nM T03917 C37YFP 44285838 IC50 = 38000 nM T03917 C9XAF7 44285850 IC50 = 77000 nM T03917 C03GEO 44285957 IC50 = 52000 nM T03917 CPL4G9 44286233 IC50 = 61000 nM T03917 CMZ6L9 44286234 IC50 = 10000 nM T03917 C2XU9Q 44302377 IC50 > 400000 nM T03917 CP7Y0U 44305318 IC50 = 1600 nM T03917 CC14YG 44305495 IC50 = 1600 nM T03917 CGA95X 44334165 IC50 = 200 nM T03917 CL67WX 44334168 IC50 = 250 nM T03917 C1H0RO 44346765 IC50 = 5000 nM T03917 C1ZY2O 44349458 IC50 = 200 nM T03917 CUM8V1 44349468 IC50 = 100 nM T03917 CK3E2P 44349473 IC50 = 160 nM T03917 CG8O0Z 44349474 IC50 = 100 nM T03917 CCQO15 44349475 IC50 = 130 nM T03917 CMVX89 44349476 IC50 = 800 nM T03917 C94GUN 44349650 IC50 = 4000 nM T03917 C1X4JZ 44349653 IC50 = 250 nM T03917 C7P9WK 44349753 IC50 = 500 nM T03917 C7TIS1 44349762 IC50 = 130 nM T03917 CO2NA8 44566805 IC50 > 150000 nM T03917 C9V3RF 44582881 IC50 = 810 nM T03917 C5SU6C 44582893 IC50 = 760 nM T03917 C6W0IC 44583703 IC50 > 100 ug.mL-1 T03917 CNU2E8 44588852 IC50 = 117000 nM T03917 CN0A6D 44588853 IC50 = 4000 nM T03917 CL40IJ 46210048 IC50 > 100000 nM T03917 C9BOT1 46905254 IC50 = 64.5 nM T03917 C50BMI 53484102 IC50 = 9000 nM T03917 CSU9E4 53484119 IC50 = 6000 nM T03917 C5JQK8 53484121 IC50 = 6000 nM T03917 CO7U4M 53494115 IC50 = 19000 nM T03917 C7JUY6 53494117 IC50 = 17000 nM T03917 CT7LC4 53494119 IC50 = 14000 nM T03917 C2IYQ6 53494251 IC50 = 18000 nM T03917 CM1D7S 56666216 IC50 = 5000 nM T03917 CE2GK6 56683110 IC50 = 8000 nM T03917 C6DSY4 60200373 IC50 = 54.1 ug.mL-1 T03917 C2UBG6 60200532 IC50 > 100 ug.mL-1 T03917 C6VJ5W 60200533 IC50 > 100 ug.mL-1 T03917 C3VWR6 60200697 IC50 > 100 ug.mL-1 T03917 CU5K4C 60200698 IC50 > 100 ug.mL-1 T03917 C6LA4B 70682440 IC50 = 2000 nM T03917 CH7FO9 70682442 IC50 = 360 nM T03917 C0OSF5 70682443 IC50 = 36000 nM T03917 CD8ZA5 70682446 IC50 = 400 nM T03917 C7LZ2Q 70682447 IC50 = 40000 nM T03917 C8WIJ2 70682448 IC50 > 100000 nM T03917 C92IFQ 70682894 IC50 = 150 nM T03917 CJMI69 70684534 IC50 = 1070 nM T03917 C4ZTH6 70684538 IC50 = 15000 nM T03917 C2K0UW 70684540 IC50 = 60 nM T03917 C37IFY 70686667 IC50 = 12500 nM T03917 C9E0QZ 70686673 IC50 > 100000 nM T03917 C7Y1GI 70688765 IC50 = 500 nM T03917 CVF5U8 70688766 IC50 = 160 nM T03917 CE4AJ1 70688769 IC50 = 7943.28 nM T03917 C4TOH1 70688907 IC50 > 100 ug.mL-1 T03917 CGXF49 70689204 IC50 = 7 nM T03917 C9KBV4 70689206 IC50 = 500 nM T03917 CSK46X 70689213 IC50 = 75 nM T03917 CJX83M 70690844 IC50 = 1000 nM T03917 CVH63D 70690845 IC50 = 20 nM T03917 CW78IM 70690846 IC50 = 30 nM T03917 C9SV7A 70690847 IC50 = 30 nM T03917 C2N1OD 70690848 IC50 = 88 nM T03917 C3PXU2 70690852 IC50 = 12 nM T03917 CZ2FQ5 70690857 IC50 = 1580 nM T03917 CUCD25 70692987 IC50 = 200 nM T03917 CKE34D 70692988 IC50 = 2000 nM T03917 C8MC2Z 70692993 IC50 > 100000 nM T03917 CM9L7V 70693001 IC50 > 100000 nM T03917 CC90RH 70693002 IC50 = 50000 nM T03917 CJF78W 70693003 IC50 = 270 nM T03917 CWAM26 70695036 IC50 = 100 nM T03917 CZ2G3A 70695039 IC50 = 45 nM T03917 CD1U7K 70695187 IC50 = 59.4 ug.mL-1 T03917 C6F5LE 70695502 IC50 = 400 nM T03917 CUQX18 70697075 IC50 = 610 nM T03917 CM0CD1 70697077 IC50 = 79000 nM T03917 C8V9WP 70697078 IC50 = 250 nM T03917 CWZ81R 70697079 IC50 = 80 nM T03917 CCD32V 70697083 IC50 = 1260 nM T03917 C50EHP 70697085 IC50 = 99 nM T03917 CE26OR 70697531 IC50 = 3 nM T03917 CU43QH 71449196 IC50 = 400 nM T03917 CT8OH3 71450945 IC50 = 1000 nM T03917 CWV76F 71459885 IC50 = 1600 nM T03917 C3Y4HN 71461587 IC50 = 3000 nM T03917 CN3QS2 73350759 IC50 > 100000 nM T03917 CX86AC 73355247 IC50 > 100000 nM T03917 C1WJ3Z 73356789 IC50 > 100000 nM T03917 C4F9ZM 73356790 IC50 > 100000 nM T03917 C4J3EO 76311384 IC50 = 2000 nM T03917 C0Q4GY 76311415 IC50 = 800 nM T03917 CQDB36 76313491 IC50 = 70 nM T03917 CB58MD 76313492 IC50 = 1300 nM T03917 C0ICG1 76313499 IC50 = 20000 nM T03917 C0WKB3 76317007 IC50 = 9 nM T03917 CGL01Q 76317008 IC50 = 8 nM T03917 CJE71Z 76317009 IC50 = 650 nM T03917 C1UXS7 76317012 IC50 = 6000 nM T03917 CEJ1O7 76318608 IC50 = 2000 nM T03917 C0AEU9 76318635 IC50 = 600 nM T03917 CG91XB 76318636 IC50 = 4500 nM T03917 CXGH63 76318652 IC50 = 10000 nM T03917 C3X0TP 76320723 IC50 = 24000 nM T03917 C8QYT7 76320724 IC50 > 200000 nM T03917 CNL6H3 76324371 IC50 = 800 nM T03917 C0Y3PQ 76325878 IC50 > 10000 nM T03917 CG6XL8 76327931 IC50 = 8 nM T03917 C6M7AP 76327932 IC50 = 650 nM T03917 C2C3FJ 76327933 IC50 = 650 nM T03917 C6G8IC 76327940 IC50 = 46000 nM T03917 CE8TP2 76331587 IC50 = 20000 nM T03917 CVGS16 76335203 IC50 = 1000 nM T03917 CN2JS0 76335217 IC50 = 6000 nM T03917 CQ20GC 86288868 IC50 = 87 nM T03917 CZ4H5C 90683388 IC50 > 150000 nM T03917 CDQ5Z7 101694272 IC50 = 10.5 nM T03917 CJ0B5W 118718121 IC50 = 12000 nM T03917 CKT3A0 118718512 IC50 = 2500 nM T03917 CTYJ95 118718769 IC50 = 10.7 nM T03917 C1XJT0 127037890 IC50 = 21.6 ug.mL-1 T03917 C8L4OC 127039260 IC50 > 128 ug.mL-1 T03917 CW62TP 127042207 IC50 = 35.8 ug.mL-1 T03917 C17XWG 127042208 IC50 = 42.5 ug.mL-1 T03917 CV9MO0 127042558 IC50 = 123.5 ug.mL-1 T03917 CF45CS 127042559 IC50 > 128 ug.mL-1 T03917 CDT2K5 132516354 IC50 > 100000 nM T03917 C6Q7BP 132516355 IC50 > 100000 nM T03917 C6THO0 139051522 IC50 > 128000 nM T03917 CC62TK 139586668 IC50 > 100000 nM T03917 CT6SE5 139587886 IC50 > 100000 nM T03917 C4NIJ3 145950197 IC50 > 128000 nM T03917 CW8K4Z 145951601 IC50 > 128000 nM T03917 C35JVR 145953467 IC50 > 100000 nM T03917 CU9X0S 145953519 IC50 > 100000 nM T03917 CXBG45 145953571 IC50 > 128000 nM T03917 C0H2KM 145959181 IC50 > 128000 nM T03917 CC6S3K 145960325 IC50 > 128000 nM T03917 CRJ1K6 145960597 IC50 > 150000 nM T03917 CGQW92 145960709 IC50 > 150000 nM T03917 CJ1OB8 145960940 IC50 > 150000 nM T03917 C96SIR 145961345 IC50 > 150000 nM T03917 C7XYJ9 145961616 IC50 > 150000 nM T03917 C75WVH 145961732 IC50 = 110000 nM T03917 C0GFZ9 145962298 IC50 > 150000 nM T03917 CO2QW3 145962675 IC50 = 120000 nM T03917 CU8LB7 145962983 IC50 > 150000 nM T03917 CMZ8D5 145971529 IC50 > 100000 nM T03917 CAG1X0 145974301 IC50 > 128000 nM T03917 CNY2L0 145982650 IC50 = 330 nM T03917 C2CEJ3 145982848 IC50 = 1140 nM T03917 C54TYD 145982890 IC50 = 450 nM T03917 CP0BZ9 145983084 IC50 = 750 nM T03917 C4XAN2 145983498 IC50 = 910 nM T03917 C1SA5K 145983558 IC50 = 770 nM T03917 CF8NB6 145983602 IC50 = 870 nM T03917 C2BZ6N 145983854 IC50 = 540 nM T03917 C8FJ9L 145984126 IC50 = 960 nM T03917 C0ZSO7 145984461 IC50 = 300 nM T03917 C5P3TX 145984503 IC50 = 1180 nM T03917 CSWO70 145984543 IC50 = 410 nM T03917 CA6NR1 145984600 IC50 = 1050 nM T03917 C5CPG1 145985072 IC50 = 1140 nM T03917 C6P0AH 145985196 IC50 = 700 nM T03917 CM5V7W 145985204 IC50 = 260 nM T03917 CGNO68 145985478 IC50 = 1180 nM T03917 CEJK76 145985579 IC50 = 360 nM T03917 CZ82FS 145985696 IC50 = 1130 nM T03917 C80FSI 145985754 IC50 = 1090 nM T03917 CVH0F6 145985890 IC50 = 1230 nM T03917 C3XN6S 145986001 IC50 = 910 nM T03917 C1M4GO 145986107 IC50 = 410 nM T03917 C5TIS2 145986169 IC50 = 1380 nM T03917 D08ZNS 4369270 IC50 = 20 nM T03917 D0M9VY 23662099 IC50 = 3000 nM T03917 D0Q4QF 6509753 IC50 > 150000 nM T37848 D00AXJ 4189 IC50 = 851.14 nM T37848 D00FGR 3599 IC50 > 100000 nM T37848 D00IBN 54676228 IC50 = 1000000 nM T37848 D00KHM 16362 IC50 = 9700 nM T37848 D00KVO 2082 IC50 > 30000 nM T37848 D00YZD 54726191 IC50 = 54000 nM T37848 D01AXB 60835 IC50 = 440 nM T37848 D01QIN 60823 IC50 = 5100 nM T37848 D01XBA 5035 Ki = 9900 nM T37848 D01XNB 4594 IC50 = 77983.01 nM T37848 D01ZII 2726 IC50 = 23300 nM T37848 D02DPA 2756 IC50 = 15000 nM T37848 D02HED 4748 IC50 = 13900 nM T37848 D02OZE 2724385 IC50 > 50000 nM T37848 D02STN 132971 IC50 = 230 nM T37848 D02VJP 25151504 IC50 = 150 nM T37848 D02YIZ 12560 IC50 = 1900 nM T37848 D03BLF 31307 IC50 = 49100 nM T37848 D03HJK 447043 IC50 > 10000 nM T37848 D03WEX 9966051 IC50 = 10000 nM T37848 D04JEE 4946 IC50 > 10000 nM T37848 D04NQI 2165 IC50 > 50000 nM T37848 D04OSE 4485 IC50 = 5620 nM T37848 D04XGT 31593 IC50 = 98200 nM T37848 D05CEU 941361 IC50 > 50000 nM T37848 D05EAM 4735 IC50 > 25000 nM T37848 D05LBU 5472 IC50 = 32700 nM T37848 D06ABF 3957 IC50 > 30000 nM T37848 D06GDY 43815 IC50 = 24100 nM T37848 D06GKN 2099 IC50 = 600 nM T37848 D06IGU 202225 IC50 = 20000 nM T37848 D06MAJ 65906 IC50 > 5000 nM T37848 D06NXY 5991 Ki = 18000 nM T37848 D06OMK 445643 IC50 = 120 nM T37848 D06XMU 6013 IC50 = 10000 nM T37848 D06YFA 31101 IC50 = 2999.16 nM T37848 D07ABV 468595 IC50 = 50 nM T37848 D07ACT 5479530 IC50 > 50000 nM T37848 D07ESC 11561674 IC50 > 10000 nM T37848 D07HOB 60838 Ki = 24000 nM T37848 D07JJS 5328 IC50 = 835603.02 nM T37848 D07KSG 2733526 Ki = 200 nM T37848 D07POC 176870 Ki = 6300 nM T37848 D07UYO 441401 IC50 > 20000 nM T37848 D08CDI 208908 Ki = 1700 nM T37848 D09DHY 6167 IC50 > 50000 nM T37848 D09EGZ 2719 IC50 = 349945.17 nM T37848 D09GOS 2812 IC50 = 20 nM T37848 D09HNR 3002190 IC50 = 11800 nM T37848 D09IPV 28417 IC50 > 30000 nM T37848 D09KTS 24821094 IC50 = 11000 nM T37848 D09LNI 3365 IC50 = 23969.8 nM T37848 D09MGR 123619 IC50 > 50000 nM T37848 D09SGV 25154714 IC50 = 7200 nM T37848 D09XQF 3767 Ki = 36000 nM T37848 D0A0OO 65016 Ki = 260 nM T37848 D0AZ3C 5291 Ki = 14300 nM T37848 D0AZ8C 5213 Ki = 32000 nM T37848 D0B4IF 456201 IC50 = 17 nM T37848 D0B7EB 36462 IC50 > 50000 nM T37848 D0C3SW 53465279 IC50 = 32400 nM T37848 D0D1AL 3559 IC50 = 8200 nM T37848 D0D4YZ 45375808 IC50 = 8400 nM T37848 D0D9FV 4601 IC50 > 30000 nM T37848 D0E6XR 3062316 Ki = 6300 nM T37848 D0E6YQ 1935 IC50 = 96900 nM T37848 D0E7PQ 5311 IC50 > 10000 nM T37848 D0EG1I 9926791 IC50 > 52000 nM T37848 D0EV8E 3198 IC50 = 430.53 nM T37848 D0F9BY 166548 IC50 > 17500 nM T37848 D0G4KG 3828 IC50 > 10000 nM T37848 D0GU4K 135413536 IC50 = 46 nM T37848 D0H0KB 5070 IC50 > 25000 nM T37848 D0H0ND 54454 IC50 > 30000 nM T37848 D0I1FQ 54671008 IC50 > 50000 nM T37848 D0I2MK 4171 IC50 > 50000 nM T37848 D0IT2G 5743 IC50 > 50000 nM T37848 D0K0TC 68617 IC50 = 800 nM T37848 D0K7WK 4595 IC50 = 11000 nM T37848 D0K8KX 5280343 IC50 = 2110 nM T37848 D0K9MY 11243969 IC50 > 50000 nM T37848 D0KR5B 5754 IC50 > 50000 nM T37848 D0L1JW 197835 Ki = 110000 nM T37848 D0N3VR 71616 IC50 = 13000 nM T37848 D0N6RF 65999 IC50 > 50000 nM T37848 D0NJ5H 11450633 IC50 < 10000 nM T37848 D0NS6H 3152 IC50 = 54680 nM T37848 D0O3OS 104850 IC50 > 20 nM T37848 D0OB1J 39186 Ki = 100 nM T37848 D0P0SZ 122262 Ki = 90 nM T37848 D0Q2PE 4539 IC50 > 50000 nM T37848 D0Q9EV 11965427 IC50 > 20000 nM T37848 D0Q9JT 4174 IC50 = 4931.74 nM T37848 D0R0FE 2520 IC50 = 4700 nM T37848 D0S5LO 25166913 IC50 > 30000 nM T37848 D0T0KA 4474 IC50 = 380 nM T37848 D0T6WN 6451164 IC50 = 2170 nM T37848 D0T8LY 1049 IC50 = 4000000 nM T37848 D0T8XB 44513473 IC50 > 10000 nM T37848 D0TG1H 3033 Ki = 1640000 nM T37848 D0U5GB 92727 Ki = 410 nM T37848 D0U6LM 4192 Ki = 2470 nM T37848 D0V3ZA 10531 IC50 = 2999.16 nM T37848 D0V7CF 5362440 IC50 = 150 nM T37848 D0V8HJ 11671467 IC50 > 50000 nM T37848 D0VG7Y 24785956 IC50 = 56000 nM T37848 D0W7WC 16220172 IC50 > 20000 nM T37848 D0W9MM 13342 IC50 = 26000 nM T37848 D0WE3O 5288826 IC50 > 50000 nM T37848 D0WI3T 441243 Ki = 170 nM T37848 D0X7DE 4449 IC50 = 15 nM T37848 D0Y4JJ 2351 IC50 = 23600 nM T37848 D0Y4QG 5388906 IC50 > 40000 nM T37848 D0Y7LD 222284 IC50 > 100000 nM T37848 D0Z1RV 135398737 IC50 = 46300 nM T37848 D0Z1ZM 84029 Ki = 5490 nM T37848 D0Z3DY 2333 IC50 = 29200 nM T37848 D0Z4EI 55245 Ki = 4700 nM T37848 D0Z4SB 3478 IC50 = 7447.32 nM T37848 D0Z7KE 3784 IC50 > 30000 nM T37848 D0ZU9R 392622 IC50 = 30 nM T37848 D00DRL 44137946 IC50 = 7100 nM T37848 D00FHR 9865515 IC50 = 570 nM T37848 D00JFE 56941241 IC50 > 20000 nM T37848 D00RYA 16750271 IC50 > 10000 nM T37848 D01DDN 56950369 IC50 > 50000 nM T37848 D01LCC 17754438 IC50 > 30000 nM T37848 D01QSG 16126898 IC50 > 30000 nM T37848 D01SJT 11713159 Ki = 12000 nM T37848 D02AAO 10368812 IC50 > 10000 nM T37848 D02AIN 122678117 IC50 > 20000 nM T37848 D02EEJ 6479267 IC50 = 58500 nM T37848 D02NNV 3038525 IC50 > 40000 nM T37848 D02QWY 24785538 IC50 = 7000 nM T37848 D03AND 11656518 IC50 > 40000 nM T37848 D03FOP 68947304 IC50 > 27000 nM T37848 D03GNI 2166 IC50 > 100000 nM T37848 D03ISJ 135564632 IC50 > 50000 nM T37848 D03LWG 53235510 IC50 > 10000 nM T37848 D03MFQ 9996409 IC50 = 48000 nM T37848 D03MYO 15981237 IC50 > 50000 nM T37848 D03QHC 49856296 Ki = 156 nM T37848 D03SQT 68234908 IC50 > 100000 nM T37848 D03WNG 73051463 IC50 = 1300 nM T37848 D04JTX 66561902 IC50 = 23000 nM T37848 D04MXN 56846693 IC50 > 10000 nM T37848 D04QZI 11340891 IC50 > 100000 nM T37848 D04TNT 46851313 IC50 > 10000 nM T37848 D04WUA 219101 IC50 > 20000 nM T37848 D05LRD 59286554 IC50 > 30000 nM T37848 D05OMT 45142457 IC50 = 11580 nM T37848 D05PZB 135398495 IC50 > 10000 nM T37848 D05UYQ 15984937 IC50 = 26000 nM T37848 D06DMQ 59472121 IC50 > 30000 nM T37848 D06EPO 11192346 IC50 > 30000 nM T37848 D06MHZ 66558287 IC50 = 170 nM T37848 D06QBY 10229498 IC50 = 25000 nM T37848 D06TKI 49857317 IC50 = 10000 nM T37848 D06TQR 76287260 IC50 > 50000 nM T37848 D06ZEO 54674461 IC50 > 50000 nM T37848 D07ARN 25182860 IC50 > 200000 nM T37848 D07HZG 11516136 IC50 > 30000 nM T37848 D07OFM 46943432 IC50 >= 33000 nM T37848 D07PNT 10433653 IC50 = 25000 nM T37848 D08AOZ 86582336 IC50 = 8500 nM T37848 D08HOM 46207586 IC50 > 30000 nM T37848 D08PMW 9951995 IC50 = 8100 nM T37848 D08SCL 46190695 IC50 = 17000 nM T37848 D08UGX 60652 IC50 = 690 nM T37848 D08VSQ 59336911 IC50 > 40000 nM T37848 D09DXX 71571306 IC50 > 100000 nM T37848 D09RII 71602803 IC50 = 12500 nM T37848 D09WYL 11634973 IC50 > 100000 nM T37848 D0B3FV 6445533 IC50 = 14000 nM T37848 D0B5HF 44476893 IC50 > 50000 nM T37848 D0BM7M 11488320 IC50 > 10000 nM T37848 D0C8DD 11552706 IC50 >= 79432.82 nM T37848 D0C9PZ 91754484 IC50 > 50000 nM T37848 D0CB2B 23653789 IC50 = 39000 nM T37848 D0CG8S 71305058 IC50 > 25000 nM T37848 D0CW8S 71657619 IC50 > 50000 nM T37848 D0D7TD 447451 IC50 = 2700 nM T37848 D0DH5X 44472635 IC50 > 100000 nM T37848 D0DK8X 50922691 IC50 = 3000 nM T37848 D0E0JO 117857370 EC50 > 100000 nM T37848 D0EB5N 25185057 IC50 = 4430 nM T37848 D0EM4S 17751090 IC50 > 25000 nM T37848 D0EY0A 42636350 IC50 > 30000 nM T37848 D0F4JK 11547499 IC50 > 30000 nM T37848 D0F4ZY 5311037 IC50 > 40000 nM T37848 D0F6YM 3035000 IC50 > 50000 nM T37848 D0FD6D 11751922 IC50 > 30000 nM T37848 D0G5XV 135565884 IC50 = 14300 nM T37848 D0G7UX 5284373 Ki = 300 nM T37848 D0G9AW 59473233 IC50 > 10000 nM T37848 D0GC5H 123879 IC50 > 30000 nM T37848 D0H0YD 32798 IC50 = 206 nM T37848 D0H6AG 51003469 IC50 = 100 nM T37848 D0H9DA 54761306 IC50 > 10000 nM T37848 D0H9SX 6914657 IC50 = 1500 nM T37848 D0HE7C 134415769 IC50 = 1600 nM T37848 D0HS5V 11234052 IC50 = 18000 nM T37848 D0I2XM 3038500 IC50 = 9300 nM T37848 D0I3LO 91933883 IC50 > 20000 nM T37848 D0I3TU 45268455 IC50 = 34000 nM T37848 D0I4PW 60164925 IC50 > 50000 nM T37848 D0IA9Y 53472683 IC50 = 24000 nM T37848 D0IQ0Z 46885626 IC50 = 15000 nM T37848 D0IZ8X 90111638 IC50 = 15000 nM T37848 D0J1HB 23063810 IC50 > 100000 nM T37848 D0JT5I 24771824 IC50 = 30000 nM T37848 D0K1EG 11508736 IC50 > 100000 nM T37848 D0K4FP 44548240 IC50 = 8000 nM T37848 D0K4JQ 57339460 IC50 > 33000 nM T37848 D0K5HI 5311424 IC50 = 4000 nM T37848 D0K7FY 72703790 IC50 > 25000 nM T37848 D0KR1N 6918653 Ki = 58000 nM T37848 D0L1GD 58282870 IC50 = 1700 nM T37848 D0L9KH 44623998 IC50 > 50000 nM T37848 D0L9QM 59568713 IC50 > 50000 nM T37848 D0M4TJ 44219292 IC50 > 50000 nM T37848 D0M6BD 16719221 IC50 > 100000 nM T37848 D0M8FD 4261 IC50 = 730 nM T37848 D0M9RQ 11697697 IC50 > 27000 nM T37848 D0MR0B 54766013 IC50 > 10000 nM T37848 D0N5KS 154104 IC50 = 9300 nM T37848 D0N6NM 71721648 IC50 > 5600 nM T37848 D0N6SO 15983988 IC50 < 10000 nM T37848 D0N8RV 9868037 Ki = 24000 nM T37848 D0O2XQ 11256587 IC50 > 6670 nM T37848 D0O7QA 46840946 IC50 > 30000 nM T37848 D0OK2N 24864821 IC50 = 4100 nM T37848 D0P0KN 16739650 IC50 > 25000 nM T37848 D0PN8H 46216796 IC50 > 5000 nM T37848 D0PW4N 6851740 IC50 = 4100 nM T37848 D0Q0AP 10409068 IC50 = 18000 nM T37848 D0Q7AG 53240420 IC50 = 17000 nM T37848 D0Q7NB 10253143 IC50 > 100000 nM T37848 D0QR5G 2355 IC50 > 10000 nM T37848 D0R3VK 42642654 IC50 > 10000 nM T37848 D0R9IU 44462758 IC50 > 25000 nM T37848 D0RL4X 45270144 IC50 > 30000 nM T37848 D0S0EQ 9951066 IC50 = 9000 nM T37848 D0S1XX 134821691 EC50 > 40000 nM T37848 D0S2PD 42634627 IC50 > 30000 nM T37848 D0S5IR 86294073 IC50 > 30000 nM T37848 D0SG7B 49831257 IC50 > 70000 nM T37848 D0SP5V 49843471 IC50 > 50000 nM T37848 D0T3DO 9867758 IC50 = 25000 nM T37848 D0T4SG 11292191 IC50 > 10000 nM T37848 D0U3EP 445154 Ki = 20000 nM T37848 D0U4FF 10437018 IC50 = 1600 nM T37848 D0U7KH 86567195 IC50 > 5000 nM T37848 D0U8QH 59239165 IC50 > 10000 nM T37848 D0UA9J 91886002 IC50 = 79000 nM T37848 D0V9VG 51049968 IC50 = 17000 nM T37848 D0VI4N 90409366 IC50 > 10000 nM T37848 D0VO0T 24800541 IC50 = 3500 nM T37848 D0W1US 1684 IC50 = 6309.57 nM T37848 D0W7HE 56649450 IC50 > 10000 nM T37848 D0W8XT 60663 IC50 = 130 nM T37848 D0W9VW 11526696 IC50 = 2400 nM T37848 D0X3OI 9883029 IC50 > 10000 nM T37848 D0X7EG 11462174 IC50 > 30000 nM T37848 D0XD4I 118502708 IC50 > 30000 nM T37848 D0XT6W 6918638 IC50 > 10000 nM T37848 D0Y1NC 148198 IC50 = 220 nM T37848 D0Y7NA 49871007 IC50 > 25000 nM T37848 D0YB2Y 42641863 IC50 >= 30000 nM T37848 D0ZE1O 9949641 IC50 > 50000 nM T37848 D0LF0O 135441202 IC50 = 26000 nM T37848 D03ZXG 118103874 IC50 = 3900 nM T37848 D04MAZ 71731606 IC50 = 46180 nM T37848 D08DMM 91799365 IC50 > 30000 nM T37848 D08SNH 71555922 IC50 = 15000 nM T37848 D0CI3E 50990953 IC50 = 22300 nM T37848 D0D3GL 137662068 IC50 > 40000 nM T37848 D0G2TX 46911228 IC50 > 5000 nM T37848 D0HG2S 86294663 IC50 = 17500 nM T37848 D0LI2I 118096900 IC50 > 30000 nM T37848 D0LU9X 74221950 IC50 > 50000 nM T37848 D0N6HP 91886057 IC50 = 5900 nM T37848 D0NJ9E 118096899 IC50 = 17800 nM T37848 D0QE8S 60197821 IC50 = 4300 nM T37848 D0QZ8K 70874141 IC50 = 700 nM T37848 D0TR9T 45256914 IC50 > 5000 nM T37848 D0W1XE 91827457 IC50 = 29430 nM T37848 D0WR7B 122650373 IC50 > 30000 nM T37848 D0ZM8H 25265637 IC50 > 20000 nM T37848 D00ZGA 9917021 Ki = 4930 nM T37848 D03EZB 9864291 IC50 = 3800 nM T37848 D03YPJ 5163 IC50 > 100000 nM T37848 D04RLX 148201 IC50 > 100000 nM T37848 D04WCI 16220188 IC50 > 29000 nM T37848 D04YHW 11406590 IC50 > 40000 nM T37848 D05FYA 3035905 IC50 = 6095.37 nM T37848 D05HIJ 135565159 IC50 = 40000 nM T37848 D05MCS 44473151 IC50 > 50 nM T37848 D06TGE 11226090 IC50 > 20 nM T37848 D06ZVC 10150497 IC50 = 33000 nM T37848 D07EBU 135565424 IC50 > 15000 nM T37848 D07GIB 11614352 IC50 = 9000 nM T37848 D07OCC 25019714 IC50 = 3800 nM T37848 D08QHS 11296282 IC50 = 7600 nM T37848 D08QTP 6478034 IC50 = 27500 nM T37848 D08SOF 5405 IC50 = 320 nM T37848 D09EVZ 507806 IC50 > 40000 nM T37848 D09GHB 11548630 IC50 > 100000 nM T37848 D09NBM 10417440 IC50 = 10000 nM T37848 D09VTB 71768520 IC50 >= 10000 nM T37848 D0A1NU 16049769 IC50 > 30000 nM T37848 D0B4TT 17747460 IC50 = 300 nM T37848 D0B7SP 11292933 IC50 = 21000 nM T37848 D0D3ZP 11167850 IC50 = 700 nM T37848 D0G6SZ 3001322 IC50 > 30000 nM T37848 D0GE2F 53354790 IC50 = 7100 nM T37848 D0H9GQ 9795276 IC50 = 1300 nM T37848 D0IP6X 219077 IC50 = 1000 nM T37848 D0L5UO 9939609 IC50 = 27000 nM T37848 D0M4LF 23649325 IC50 = 20000 nM T37848 D0N8NK 11641563 IC50 > 10000 nM T37848 D0N8XL 46862685 IC50 = 2000 nM T37848 D0R7GH 9833312 IC50 = 56.23 nM T37848 D0SX7F 60876 Ki = 28 nM T37848 D0Y2HR 2247 IC50 = 10600 nM T37848 D0YE2N 73214 IC50 > 20000 nM T37848 C6OZ1C 1267 IC50 = 600 nM T37848 CA28EH 1390 IC50 = 2697739.43 nM T37848 C4PZ9H 3444 IC50 = 130 nM T37848 CY4WG9 3793 IC50 = 32.6 nM T37848 C9LCD8 3823 IC50 = 1 nM T37848 C2KJI7 3883 IC50 > 30000 nM T37848 C93BJO 5039 IC50 > 50000 nM T37848 C12ETD 5380 IC50 = 289734.36 nM T37848 C65GNV 7971 IC50 = 767361.49 nM T37848 C1OVB9 12749 IC50 = 1253141.17 nM T37848 CN0WP7 15630 IC50 = 10000 nM T37848 C8B1ZX 36284 Ki = 20000 nM T37848 C5OVQ6 39385 IC50 = 9289.66 nM T37848 C6GN7M 40692 IC50 = 667 nM T37848 CN5S8L 43234 IC50 = 1039.92 nM T37848 CK6VT0 60923 IC50 = 5.8 nM T37848 CP8F7B 64143 Ki = 480 nM T37848 C2FVG0 64149 IC50 > 30000 nM T37848 CPW9G5 65126 Ki = 4300 nM T37848 CL15AQ 65373 IC50 = 47300 nM T37848 CPW9B5 65752 Ki = 107700 nM T37848 CA02CO 65808 Ki = 5100 nM T37848 CMLI08 68079 IC50 > 10000 nM T37848 C95JWC 68487 IC50 = 64700 nM T37848 CL86ZR 72171 IC50 = 309029.54 nM T37848 C4GBJ1 72310 IC50 = 30600 nM T37848 CO0HB3 75473 Ki > 400000 nM T37848 CAF69U 81130 IC50 = 430526.61 nM T37848 C7SXL6 87152 IC50 > 25000 nM T37848 C2HFT4 91673 IC50 = 210 nM T37848 C1CWL8 92305 Ki = 1390 nM T37848 C1IV2T 93168 Ki = 7930 nM T37848 CC0P7F 94378 IC50 > 30000 nM T37848 CZB67X 98608 IC50 > 10000 nM T37848 CH50RJ 104956 IC50 = 45 nM T37848 C52FVK 104972 Ki = 2110 nM T37848 C0K7OY 108137 IC50 = 12000 nM T37848 CEP43C 122068 IC50 = 24000 nM T37848 CD1JI7 124052 Ki = 7000 nM T37848 C6QB9N 126266 IC50 = 50000 nM T37848 CF0NI9 151529 Ki = 399 nM T37848 CM2H7V 152430 IC50 > 10000 nM T37848 CL54TG 160521 IC50 > 100000 nM T37848 CK8RD5 168114 IC50 = 8100 nM T37848 CJ34CF 168115 IC50 = 7100 nM T37848 CDB9P5 170922 IC50 > 25000 nM T37848 C3O4NA 179651 Ki = 23200 nM T37848 CA91IX 185559 IC50 > 80000 nM T37848 C1R6GB 189060 IC50 > 10000 nM T37848 CH0ZD7 207299 IC50 = 15000 nM T37848 CAM18T 332425 IC50 = 13700 nM T37848 C9DG0W 332427 IC50 = 25600 nM T37848 CAS18T 359052 IC50 > 30000 nM T37848 CNJU05 397855 Ki = 80 nM T37848 CDU5O6 421105 IC50 = 1000 nM T37848 CLD6J9 441074 IC50 = 28000 nM T37848 C5Q8IX 457194 IC50 = 200 nM T37848 C2K7AC 465996 IC50 = 800 nM T37848 CXH7Y0 471430 IC50 = 15000 nM T37848 C1IK6G 471500 IC50 = 2300 nM T37848 CMGZ52 471501 IC50 = 9600 nM T37848 C7HEM8 471507 IC50 = 120000 nM T37848 C6GNY7 471510 IC50 = 35000 nM T37848 CVH49X 480768 IC50 > 20000 nM T37848 CRH1D7 491206 IC50 = 400 nM T37848 C3Q0TX 493820 IC50 = 310 nM T37848 CUO16L 493830 IC50 30 nM T37848 CKC8U4 507751 IC50 = 18000 nM T37848 CPXL01 507783 IC50 > 40000 nM T37848 CM40AT 507791 IC50 > 40000 nM T37848 C18QJF 515047 IC50 = 8100 nM T37848 CEN81S 515051 IC50 = 2500 nM T37848 CHX85A 515052 IC50 = 10000 nM T37848 C2Y4TD 577307 IC50 = 1400 nM T37848 C6R5XN 595145 IC50 = 57000 nM T37848 CVRM18 595254 Ki = 28000 nM T37848 CR98MZ 613528 IC50 > 30000 nM T37848 C4FC1N 626798 IC50 > 50000 nM T37848 CX5V2H 636822 IC50 = 92300 nM T37848 CHV1X7 638701 IC50 = 570 nM T37848 CTGL43 672443 IC50 = 50000 nM T37848 CZ96AU 673837 Ki < 50000000 nM T37848 CT3J9U 673847 Ki < 50000000 nM T37848 CVM04E 675159 Ki < 50000000 nM T37848 C76MVW 675233 Ki < 50000000 nM T37848 CP8TY1 678717 Ki < 50000000 nM T37848 CGL5R1 683949 IC50 > 3750 nM T37848 CN5CJ7 688803 IC50 > 10000 nM T37848 C2AHB4 689051 IC50 > 10000 nM T37848 C74MRA 702869 IC50 = 8860 nM T37848 CQ42OY 739374 IC50 > 15000 nM T37848 C6DJ3Y 741004 IC50 = 4860 nM T37848 C8Y3TW 745415 Ki = 4100 nM T37848 C4V6EW 747770 IC50 = 34000 nM T37848 CSUL21 780263 IC50 = 12300 nM T37848 CP23UY 780805 IC50 > 30000 nM T37848 C4WCL7 792361 IC50 > 10000 nM T37848 CI43WJ 802727 IC50 > 10000 nM T37848 C3LM4S 821286 IC50 = 6000 nM T37848 C06WCN 827839 IC50 = 4230 nM T37848 CY3N7H 851298 IC50 > 39810.72 nM T37848 C1T6CV 854051 IC50 = 5000000 nM T37848 CYKE37 863679 IC50 > 20000 nM T37848 CLJU94 877119 IC50 = 10200 nM T37848 C2TDG1 883547 IC50 > 40000 nM T37848 C2FPN5 936091 IC50 = 28000 nM T37848 CMO9N5 970725 IC50 > 30000 nM T37848 C2DYP4 1035332 Ki = 3100 nM T37848 CZG18E 1201554 Ki = 22900 nM T37848 CAZT67 1283333 IC50 = 251.19 nM T37848 CV0Q3D 1302369 IC50 > 30000 nM T37848 C5G4FA 1394668 IC50 > 30000 nM T37848 CMU8T3 1410239 IC50 = 1300 nM T37848 C3KGN0 1475789 IC50 > 20000 nM T37848 CP3F4T 1476707 IC50 > 40000 nM T37848 CW4YO2 1480806 IC50 = 33000 nM T37848 C0GE2X 1619763 IC50 = 16440 nM T37848 C21HKV 1941609 IC50 > 30000 nM T37848 C3LSW0 2088634 IC50 > 50000 nM T37848 CMZG42 2133890 Ki = 14400 nM T37848 CZL8R3 2187415 IC50 > 50000 nM T37848 CP53EV 2350190 IC50 = 1900 nM T37848 CRD18Y 2407524 IC50 = 38300 nM T37848 CJ1LK6 2568387 IC50 = 1000 nM T37848 CQTY36 2650025 IC50 = 27100 nM T37848 CZY89U 2727594 IC50 = 71000 nM T37848 CD28JA 2735964 IC50 > 25000 nM T37848 C5T3HX 2748785 IC50 > 10000 nM T37848 C0ZI1F 2756534 IC50 = 3500 nM T37848 CT6P3F 2782903 IC50 = 2000 nM T37848 CF2N8O 2794167 IC50 > 30000 nM T37848 CMRX81 2811640 IC50 = 7000 nM T37848 C8PYB6 2858523 IC50 = 3000 nM T37848 CJ7UK3 2902946 Ki < 50000000 nM T37848 CTBC06 2941086 IC50 > 10000 nM T37848 C14NBG 3008866 IC50 > 40000 nM T37848 C4XNG5 3012020 IC50 = 24000 nM T37848 C6TO5V 3012027 IC50 = 10000 nM T37848 CCQI26 3012527 IC50 = 3610 nM T37848 CM70GI 3013843 IC50 = 8800 nM T37848 CQ2SG0 3031421 IC50 > 20000 nM T37848 CDF6W2 3035604 IC50 = 25000 nM T37848 CSHC84 3036172 Ki = 2600 nM T37848 CAJQ53 3040177 Ki = 70000 nM T37848 C82XOE 3083746 IC50 = 28700 nM T37848 C3GSR4 3114841 IC50 = 7700 nM T37848 C3F0GS 3120536 IC50 = 4700 nM T37848 CFPR85 3213696 IC50 = 2000 nM T37848 C2L9IF 3296768 IC50 = 9600 nM T37848 CI30FE 3463042 IC50 > 40000 nM T37848 CZN5B8 3477788 IC50 = 100 nM T37848 CSW59H 3718258 IC50 > 100000 nM T37848 CXR4Y7 3811929 IC50 = 1300 nM T37848 CK93HP 3844414 IC50 = 1600 nM T37848 CO23EI 3959338 IC50 > 20000 nM T37848 CYVR59 3989497 IC50 > 10000 nM T37848 CEP9D5 4048115 IC50 = 13000 nM T37848 CG8A3J 4193543 IC50 = 71 nM T37848 C70BNQ 4221718 Ki = 3970 nM T37848 CIF8G9 4261503 IC50 = 12000 nM T37848 CBN96T 4358655 IC50 = 1000 nM T37848 C1ZC4D 4384047 IC50 > 80 nM T37848 CBSM52 4450788 IC50 = 230 nM T37848 C7RPL4 4450789 IC50 = 26000 nM T37848 CE0OD3 4652320 IC50 > 40000 nM T37848 CZO2E5 4674678 IC50 = 4010 nM T37848 CFL8J3 4786512 IC50 = 20 nM T37848 CI4DE0 4803142 IC50 = 750 nM T37848 CBFV62 4817293 IC50 = 50000 nM T37848 CIN5F7 4904109 IC50 > 30000 nM T37848 C16EGI 4961254 IC50 > 10000 nM T37848 C7CNQ4 5201490 IC50 > 40000 nM T37848 C80NAU 5273742 IC50 = 30000 nM T37848 CZM7D8 5281794 IC50 = 8300 nM T37848 CO16PV 5282545 IC50 = 16000 nM T37848 C6C0UY 5282549 IC50 = 1000 nM T37848 CA5D1J 5289110 IC50 > 20000 nM T37848 CZ09MD 5299617 IC50 = 14600 nM T37848 CMBL90 5300578 IC50 > 20000 nM T37848 CC49SG 5316673 IC50 > 100000 nM T37848 CA7UL5 5329333 IC50 > 50000 nM T37848 COQ41S 5329336 IC50 > 100000 nM T37848 COJI90 5338258 IC50 > 10000 nM T37848 CWFP51 5338324 IC50 > 10000 nM T37848 CN0R5K 5352001 IC50 = 21800 nM T37848 C5Z0HQ 5355549 IC50 = 11100 nM T37848 C1D0RN 5470187 IC50 = 21800 nM T37848 C7IKS9 5470829 IC50 = 64863443.35 nM T37848 CUL7A5 5471349 IC50 = 2420 nM T37848 C3DU9C 5481663 IC50 > 80000 nM T37848 CB4A3U 5481990 Ki = 7500 nM T37848 C3Q2XB 5495793 IC50 > 40000 nM T37848 C0ZAM9 5495818 IC50 > 40000 nM T37848 CPT10H 5717399 IC50 = 12000 nM T37848 C21EJH 5717404 IC50 = 53000 nM T37848 CE9KZ5 5720628 IC50 = 11000 nM T37848 CJMQ48 5737900 IC50 > 20000 nM T37848 CSH9C1 5787676 IC50 > 20000 nM T37848 CMWC08 5837372 IC50 > 10000 nM T37848 CAJK62 5859537 IC50 > 20000 nM T37848 CX23PO 6020016 IC50 > 10000 nM T37848 C2V8QP 6174007 IC50 = 1520 nM T37848 CTG9I2 6258621 IC50 = 1280 nM T37848 CR8P9W 6262995 IC50 > 10000 nM T37848 CA74LD 6320546 IC50 > 30000 nM T37848 CBC0J5 6418797 IC50 = 14000 nM T37848 CGJ16S 6436013 IC50 > 5000 nM T37848 C9V5HZ 6440498 Ki = 5560 nM T37848 CB75NI 6479949 IC50 = 12300 nM T37848 C09BQE 6479956 IC50 = 30000 nM T37848 CEL6U1 6479971 IC50 = 30000 nM T37848 CGL87W 6483572 IC50 > 25000 nM T37848 CC6U7A 6493950 IC50 < 1000 nM T37848 CN0VB3 6914627 IC50 > 30000 nM T37848 C80XWJ 6914629 IC50 > 30000 nM T37848 C0QCK1 6918455 IC50 = 40000 nM T37848 CP8T7C 7017202 IC50 = 1500 nM T37848 C48OIX 7074967 Ki > 400000 nM T37848 CU68IK 7141881 IC50 > 10000 nM T37848 CWX15G 7514880 IC50 = 15000 nM T37848 CJH57U 8854335 IC50 = 18000 nM T37848 C2W6PI 8867347 IC50 > 15000 nM T37848 C5J8HN 8902499 IC50 > 20000 nM T37848 C24MJV 9554928 IC50 = 33200 nM T37848 C32HVW 9554933 IC50 > 100000 nM T37848 CIA9B5 9794218 IC50 > 100000 nM T37848 CA15IT 9796590 IC50 > 10000 nM T37848 CUGX54 9797385 IC50 > 25000 nM T37848 CVZG73 9799417 IC50 > 200000 nM T37848 CBED14 9799604 IC50 = 19000 nM T37848 C7KR1T 9799867 IC50 = 2500 nM T37848 C5KZ9F 9805776 IC50 = 46000 nM T37848 CMIW83 9812710 IC50 > 30000 nM T37848 CR8ET5 9814387 IC50 = 16000 nM T37848 CFW74D 9815391 IC50 > 100000 nM T37848 CTN13P 9820134 IC50 > 100000 nM T37848 C1E2DV 9826083 IC50 > 2000 nM T37848 CRU16A 9827020 IC50 = 6.3 nM T37848 C32UFI 9828452 IC50 = 30150 nM T37848 C3NO4W 9828630 IC50 = 11.5 nM T37848 C7GSI3 9830209 Ki = 820 nM T37848 CRQA29 9830290 IC50 < 1000 nM T37848 C4TB5Y 9831072 IC50 = 8000 nM T37848 C2XA5B 9835305 IC50 > 30000 nM T37848 CJDP76 9838675 EC50 = 5900 nM T37848 CA6N0H 9843867 IC50 = 8900 nM T37848 C7VSU2 9845018 IC50 = 1000 nM T37848 CL79YZ 9858476 IC50 = 9100 nM T37848 CAQ52K 9861918 IC50 = 6700 nM T37848 CAOK24 9867098 IC50 = 6600 nM T37848 C74JKE 9868115 IC50 = 7000 nM T37848 CI6V2U 9870337 IC50 = 350 nM T37848 CQ4LC2 9872676 IC50 > 30000 nM T37848 CTZP28 9875352 IC50 = 10 nM T37848 CBF9T3 9879532 IC50 = 6800 nM T37848 CUK64X 9880846 IC50 > 10000 nM T37848 CQHE82 9883170 IC50 = 2100 nM T37848 C8YQ6V 9883171 IC50 = 5300 nM T37848 CJW1P5 9888494 IC50 > 100000 nM T37848 C9C8JK 9890681 IC50 = 9700 nM T37848 CFZ27W 9894997 IC50 = 4000 nM T37848 CJ56EL 9904146 IC50 = 1200 nM T37848 CUZT98 9906455 IC50 = 9300 nM T37848 C4B2QY 9913339 IC50 = 13000 nM T37848 C4PF5A 9923132 IC50 > 10000 nM T37848 C29WVT 9923385 IC50 > 25000 nM T37848 C3TH4Q 9927224 IC50 = 3600 nM T37848 C9FZO7 9932679 IC50 = 5000 nM T37848 CGL13H 9939495 IC50 = 11000 nM T37848 CFC48H 9940105 IC50 = 430 nM T37848 CEB1I2 9945500 IC50 > 25000 nM T37848 C9S0AG 9948129 IC50 < 1000 nM T37848 CG9KR4 9948238 IC50 > 20000 nM T37848 C8RPF6 9949067 IC50 = 2000 nM T37848 CPG94B 9952648 IC50 = 4300 nM T37848 CNJ81W 9959174 IC50 = 11000 nM T37848 CO87YK 9961741 IC50 = 4 nM T37848 C3IQV6 9965885 IC50 > 10000 nM T37848 CKLH03 9967123 IC50 = 22000 nM T37848 CISM03 9976141 IC50 = 58000 nM T37848 CJOV70 9983904 IC50 = 26000 nM T37848 CGEJ24 9985625 IC50 = 39000 nM T37848 C98KZE 10002960 IC50 = 1700 nM T37848 C26QHZ 10005638 IC50 > 2000 nM T37848 CCD24K 10007859 IC50 >= 18000 nM T37848 C1F2RH 10008768 IC50 = 7500 nM T37848 C0KHW3 10022393 IC50 = 66500 nM T37848 C5TRX2 10025406 IC50 = 5000 nM T37848 CA06TQ 10028888 IC50 > 100000 nM T37848 CQI0Z7 10029563 IC50 = 9730 nM T37848 C47DPZ 10030750 IC50 = 30000 nM T37848 C0HN4T 10031184 IC50 = 42260 nM T37848 C1WH8Q 10042344 IC50 > 40000 nM T37848 CGNA89 10045603 IC50 = 75000 nM T37848 C4SON9 10046844 IC50 < 1000 nM T37848 CPI2Q0 10049358 IC50 = 38000 nM T37848 C1DB0X 10055750 IC50 = 10000 nM T37848 CSOR04 10070428 IC50 = 51000 nM T37848 C5B4HJ 10071498 IC50 > 100000 nM T37848 CL8WC4 10075685 IC50 > 30000 nM T37848 CVE2T1 10076176 IC50 = 3800 nM T37848 CR01QE 10076802 IC50 = 20000 nM T37848 CSY53V 10077700 IC50 = 24000 nM T37848 CJO8N5 10088963 IC50 = 85600 nM T37848 C1XH8C 10091613 IC50 = 1820 nM T37848 C2G3MJ 10099429 IC50 > 30000 nM T37848 CEA01V 10108128 IC50 = 4460 nM T37848 CVK61T 10116047 IC50 = 1.4 nM T37848 C1TY3F 10122289 IC50 = 5000 nM T37848 C0KOC5 10122452 IC50 = 29000 nM T37848 C1LSI8 10122657 IC50 = 10000 nM T37848 CC2YT5 10122981 IC50 = 5200 nM T37848 CLM97C 10123174 IC50 = 50 nM T37848 C6HR7P 10130125 IC50 > 100000 nM T37848 C47RHT 10130685 IC50 = 50000 nM T37848 CD75GU 10131619 IC50 > 10000 nM T37848 CRW07C 10133485 IC50 > 50000 nM T37848 CP64RT 10134089 IC50 > 10000 nM T37848 CXS21P 10142377 IC50 = 22000 nM T37848 CR6H9Y 10146899 IC50 = 320 nM T37848 COFT51 10154555 IC50 > 100000 nM T37848 CQO8H3 10157813 IC50 > 30000 nM T37848 C1VQ4M 10162564 IC50 > 10000 nM T37848 CLT63F 10166543 IC50 = 41000 nM T37848 CJ4R2U 10168216 IC50 = 18000 nM T37848 CP6Q1W 10173403 IC50 = 58000 nM T37848 C4Z3IS 10175330 IC50 = 700 nM T37848 C6OH0I 10184529 IC50 = 15000 nM T37848 CFUO45 10184774 IC50 = 44000 nM T37848 CJ1O9P 10185917 IC50 = 8300 nM T37848 CAK3E1 10189993 IC50 = 5000 nM T37848 CDP14A 10190433 IC50 = 400 nM T37848 CEDW91 10190506 IC50 = 500 nM T37848 CA4N2V 10198034 IC50 > 100000 nM T37848 CM0F5B 10198293 IC50 = 70600 nM T37848 CG6IF7 10212348 IC50 = 1500 nM T37848 CJQU63 10212550 IC50 = 80 nM T37848 C8DWX5 10219789 IC50 > 100000 nM T37848 C5LM9R 10221470 IC50 > 125000 nM T37848 CX32UD 10223809 IC50 > 100000 nM T37848 CV5X8A 10224181 IC50 > 2500 nM T37848 C4JN9U 10224745 IC50 > 50000 nM T37848 C3FN5E 10226546 IC50 = 100000 nM T37848 CFQ5L2 10232552 IC50 = 13000 nM T37848 CB72SI 10233112 IC50 = 17000 nM T37848 C9UIX5 10233517 IC50 = 15000 nM T37848 C1B7ZE 10233723 IC50 = 480 nM T37848 CKE5C6 10233724 IC50 = 2200 nM T37848 C3OE5Z 10257392 IC50 = 19000 nM T37848 C4KU1Y 10268204 IC50 > 25000 nM T37848 CU1ZW4 10268255 IC50 = 5100 nM T37848 C2EO1A 10273854 IC50 = 27000 nM T37848 C5Z2IG 10278742 IC50 = 1000 nM T37848 CE9ID0 10280944 IC50 = 9300 nM T37848 C61ZEV 10282620 IC50 = 7000 nM T37848 CWOR29 10283706 IC50 = 440 nM T37848 CO38FQ 10283896 IC50 = 5000 nM T37848 C16MNJ 10284289 IC50 < 1000 nM T37848 CO2LT5 10286610 IC50 > 40000 nM T37848 C7C5FN 10294289 IC50 < 1000 nM T37848 CE4Y7G 10294290 IC50 > 30000 nM T37848 C3FL9K 10295633 IC50 > 2000 nM T37848 C7SFI1 10296883 Ki = 2900 nM T37848 CO0P4F 10301330 IC50 = 19700 nM T37848 CU13DH 10304547 Ki = 23000 nM T37848 CQV98P 10305047 IC50 = 22000 nM T37848 C7W2NF 10305573 IC50 = 39000 nM T37848 C9C3KH 10305705 IC50 = 310 nM T37848 CAU47H 10305883 IC50 = 110 nM T37848 CD3ER5 10308589 IC50 > 50000 nM T37848 C6ITS2 10313487 IC50 > 100000 nM T37848 CZ18PL 10316203 IC50 > 100000 nM T37848 C8F1LK 10318708 IC50 = 65000 nM T37848 C27TCH 10319351 IC50 = 6000 nM T37848 CQT7H4 10320818 IC50 = 1360 nM T37848 CM46XO 10327211 IC50 = 300 nM T37848 CEMU16 10335364 IC50 > 10000 nM T37848 C4AJ0X 10341839 IC50 > 100000 nM T37848 CFXA48 10343679 IC50 > 25000 nM T37848 CW50TU 10345610 IC50 > 30000 nM T37848 CQVP17 10347783 IC50 = 14000 nM T37848 CPD85J 10347896 IC50 > 30000 nM T37848 CH38EM 10353296 IC50 > 100000 nM T37848 C6QTS1 10358881 IC50 > 2500 nM T37848 CW9P2U 10364379 IC50 = 82000 nM T37848 CDA5F7 10369999 IC50 = 17000 nM T37848 C4A5SP 10379988 IC50 > 10000 nM T37848 C07XHY 10388612 IC50 = 5100 nM T37848 CA8B5T 10390073 IC50 > 2000 nM T37848 CJQV19 10391684 IC50 = 830 nM T37848 C0EQX7 10394458 IC50 = 180 nM T37848 CE0AS5 10405951 IC50 = 30000 nM T37848 CWK4O1 10406239 IC50 >= 5000 nM T37848 C8K7VS 10410589 IC50 = 68000 nM T37848 CH70EY 10414856 IC50 = 80 nM T37848 CR1YG5 10415353 IC50 = 39000 nM T37848 CBN4H0 10415698 IC50 = 4700 nM T37848 C0YSQ7 10416713 IC50 = 450 nM T37848 C18MRG 10436237 IC50 = 30000 nM T37848 C2O1EQ 10438856 IC50 = 800 nM T37848 C97LHV 10454092 IC50 < 100 nM T37848 C9ODF7 10454589 IC50 = 85400 nM T37848 CW4BK0 10455921 IC50 = 45800 nM T37848 C8DWH6 10456892 IC50 > 30000 nM T37848 C25FVM 10457343 IC50 = 23000 nM T37848 C1H5RP 10458842 IC50 > 10000 nM T37848 CFIE04 10459196 IC50 = 20600 nM T37848 CGXY36 10482372 IC50 = 28000 nM T37848 CHNT90 10483685 IC50 = 2500 nM T37848 C8TPU0 10510985 Ki = 251000 nM T37848 C4CRA8 10624340 IC50 = 90000 nM T37848 C6UX4J 10633725 IC50 > 10000 nM T37848 CAC8P4 10647667 IC50 = 77600 nM T37848 CJPW17 10654534 Ki > 400000 nM T37848 CQSJ50 10692619 IC50 = 73500 nM T37848 CA82YQ 10704488 IC50 > 20000 nM T37848 CXK63D 10829689 IC50 = 40300 nM T37848 CBK06L 10861643 IC50 = 81000 nM T37848 CZS9Q5 10899427 IC50 = 23900 nM T37848 CD10XK 10928028 IC50 = 2800 nM T37848 CH61UW 11128957 IC50 > 20000 nM T37848 CW1Q6S 11148656 IC50 = 58100 nM T37848 CCD91J 11148936 IC50 = 50900 nM T37848 CXT8Y2 11151568 IC50 < 10000 nM T37848 C4HBU9 11153488 IC50 = 630 nM T37848 CB47FY 11154357 IC50 > 100000 nM T37848 CKPQ58 11154980 IC50 = 4 nM T37848 C3X0AC 11155482 IC50 = 65000 nM T37848 C1R4CH 11158071 IC50 = 370 nM T37848 C5K4PC 11160258 IC50 > 100000 nM T37848 C5E8LY 11168500 IC50 = 200 nM T37848 C1A8HL 11171679 Ki = 147000 nM T37848 CP1EI3 11172276 IC50 = 9170 nM T37848 CJEW09 11176034 IC50 > 50000 nM T37848 C84PJK 11177283 IC50 = 19300 nM T37848 CYQ98P 11179994 IC50 = 15000 nM T37848 CRU5Y3 11183547 IC50 > 100000 nM T37848 CY57GR 11187635 IC50 > 50000 nM T37848 CYB1W9 11187925 IC50 = 14700 nM T37848 C0XCD3 11195292 IC50 = 44300 nM T37848 C7F6CE 11195591 IC50 = 93800 nM T37848 CHM83A 11199490 IC50 = 19200 nM T37848 C8CWV4 11200621 IC50 = 9250 nM T37848 C6XUE4 11201011 IC50 > 100000 nM T37848 CP3D7X 11201812 IC50 = 300 nM T37848 C7U4SP 11203112 IC50 = 55800 nM T37848 C9M4JX 11203238 IC50 = 4400 nM T37848 C27OAY 11204336 IC50 = 35 nM T37848 CTS40R 11204595 IC50 = 17000 nM T37848 C1XR3I 11206290 Ki = 29400 nM T37848 CJ1O6V 11207072 IC50 = 75100 nM T37848 CV1SD9 11208566 IC50 > 10000 nM T37848 CLT87I 11212921 IC50 = 9440 nM T37848 CD8VO1 11214464 IC50 = 18480 nM T37848 C4O3QM 11218177 IC50 = 7520 nM T37848 CIB34F 11218910 IC50 = 62500 nM T37848 CI2SN0 11222420 IC50 > 25000 nM T37848 C71YJO 11223701 IC50 = 20000 nM T37848 CF3AY1 11225369 IC50 = 10 nM T37848 CP9Z1V 11225445 IC50 = 440 nM T37848 C63QRZ 11226516 IC50 = 20030 nM T37848 CEW9L6 11228293 Ki = 66 nM T37848 CMHY80 11229234 Ki > 400000 nM T37848 CA71OC 11235004 IC50 > 100000 nM T37848 C9WY6K 11235389 IC50 > 50000 nM T37848 CVO5A3 11235737 IC50 = 1590 nM T37848 C6D3UR 11237434 IC50 > 30000 nM T37848 C8IQ7N 11247557 IC50 = 57000 nM T37848 C79PBA 11247947 IC50 = 2530 nM T37848 CB68XN 11249025 IC50 = 1200 nM T37848 C86MWN 11249529 IC50 = 5780 nM T37848 CLR09Q 11253245 IC50 > 100000 nM T37848 COW4I8 11259499 IC50 = 250 nM T37848 CY10OR 11260438 IC50 > 100000 nM T37848 CEN76W 11261262 IC50 = 11790 nM T37848 CD7J9T 11262242 IC50 = 8200 nM T37848 C7KU1G 11264664 IC50 > 100000 nM T37848 C92CYH 11265950 IC50 > 10000 nM T37848 CI1M9O 11270541 IC50 = 53810 nM T37848 CP13GR 11270563 IC50 = 6620 nM T37848 C9W2NY 11274374 Ki = 18 nM T37848 C9W4KE 11275964 IC50 = 883 nM T37848 CT4IL9 11281280 IC50 = 1900 nM T37848 CY79US 11293906 IC50 = 1230 nM T37848 CFX64S 11293909 IC50 = 26410 nM T37848 CH7E1O 11293927 IC50 > 100000 nM T37848 C1YH6T 11295806 IC50 = 33690 nM T37848 CQ2AW4 11299991 IC50 = 98200 nM T37848 CB0UJ7 11302765 IC50 = 8700 nM T37848 CJYA49 11304370 IC50 = 17850 nM T37848 CBEW43 11308052 IC50 = 5000 nM T37848 CF5YS9 11310529 Ki = 110000 nM T37848 CK8L6D 11310871 IC50 = 35500 nM T37848 CB7YS1 11315814 IC50 = 3300 nM T37848 C8S4FU 11317045 IC50 > 29100 nM T37848 CO8B7R 11317439 IC50 >= 1000 nM T37848 CMQD35 11321674 Ki > 400000 nM T37848 C7WA0E 11322127 IC50 = 51100 nM T37848 CY9KM7 11322128 IC50 > 100000 nM T37848 CT6CH4 11322177 IC50 = 26800 nM T37848 CW01KR 11322201 IC50 > 100000 nM T37848 C95WQP 11326501 IC50 = 1600 nM T37848 C0B2FT 11327284 IC50 = 100 nM T37848 CL8ZT6 11327691 IC50 = 1530 nM T37848 C19BEF 11330998 IC50 = 82 nM T37848 C74LWO 11331001 IC50 = 36000 nM T37848 CU72EY 11344157 Ki = 131000 nM T37848 CPK71M 11345209 IC50 > 100000 nM T37848 C2SN5F 11354531 IC50 = 2300 nM T37848 C5FG8X 11355925 IC50 > 400000 nM T37848 C84IUF 11357143 IC50 = 42600 nM T37848 C7I4FX 11363702 IC50 > 10000 nM T37848 C54CWH 11364404 IC50 = 5300 nM T37848 C7DUQ5 11364979 IC50 = 14400 nM T37848 CT6MO8 11365653 IC50 = 28000 nM T37848 CGW8R0 11366073 IC50 = 13000 nM T37848 C8N0GX 11368215 IC50 = 116 nM T37848 CI5GZ4 11368318 IC50 = 48400 nM T37848 C31PLX 11376266 IC50 = 31310 nM T37848 CC0L7O 11377200 IC50 = 7000 nM T37848 C18WDP 11377534 IC50 = 7200 nM T37848 C1BOK3 11378800 Ki < 25000 nM T37848 C0YO8L 11378954 IC50 > 100000 nM T37848 CD82VI 11379226 IC50 > 100000 nM T37848 CD68AR 11380674 IC50 < 50 nM T37848 CDF21W 11387864 IC50 = 12 nM T37848 CGY80S 11388586 IC50 = 5500 nM T37848 CZIC23 11389737 IC50 = 114000 nM T37848 CYL06Q 11389927 IC50 = 39100 nM T37848 CKZV96 11393842 IC50 = 54200 nM T37848 C9AOM3 11397017 IC50 > 10000 nM T37848 C5VC8J 11406760 IC50 = 1835 nM T37848 CWX2P1 11406781 IC50 = 1800 nM T37848 C0G4AF 11408751 IC50 > 100000 nM T37848 CIA75B 11410766 IC50 = 800 nM T37848 CUO79V 11419244 IC50 > 100000 nM T37848 C5VG6X 11421025 IC50 = 3000 nM T37848 CSU47B 11421412 IC50 = 230 nM T37848 C1V7WT 11422288 IC50 = 14 nM T37848 CLR3W7 11424804 IC50 = 22900 nM T37848 CUSQ84 11430331 IC50 > 100000 nM T37848 CFTC85 11432169 IC50 = 130 nM T37848 C0PWX2 11441615 IC50 = 2032 nM T37848 C1YV6P 11442292 IC50 > 100000 nM T37848 CTK09U 11443156 IC50 = 36820 nM T37848 CLB97A 11443942 IC50 = 8100 nM T37848 CM2J9W 11444700 IC50 = 2440 nM T37848 C62PUD 11445240 IC50 = 5000 nM T37848 C3CU1H 11450354 IC50 > 40000 nM T37848 CSK8F9 11453657 IC50 > 100000 nM T37848 CE42DM 11453673 IC50 > 100000 nM T37848 C19WQH 11454150 IC50 = 1790 nM T37848 CTQS76 11454703 IC50 = 20800 nM T37848 CYCB17 11455462 IC50 > 100000 nM T37848 C5CGK7 11456285 IC50 = 48000 nM T37848 CPIH90 11458616 IC50 > 100000 nM T37848 CIDT15 11464169 IC50 = 1400 nM T37848 CR4N5I 11465834 IC50 = 5000 nM T37848 CDZ53U 11467552 IC50 = 15848.93 nM T37848 C16NBP 11467753 IC50 = 6000 nM T37848 C9S0ZO 11474913 IC50 = 200 nM T37848 C2KXN4 11475327 IC50 = 2010 nM T37848 CW57BU 11480732 IC50 = 79200 nM T37848 CJ14TI 11485574 IC50 = 120000 nM T37848 CH0T1B 11488138 IC50 > 100000 nM T37848 COC7Q9 11488952 IC50 = 2500 nM T37848 CV5I3W 11490693 IC50 = 31800 nM T37848 C1O9XD 11493620 IC50 > 10000 nM T37848 CW3YO5 11494768 IC50 > 50000 nM T37848 CXW96U 11495012 IC50 = 1000 nM T37848 C39PJT 11495962 IC50 = 10 nM T37848 CL17QT 11497455 IC50 > 10000 nM T37848 CDM39K 11497693 IC50 = 2.3 nM T37848 C69AMJ 11500781 IC50 > 10000 nM T37848 CEV5B3 11501485 IC50 = 700 nM T37848 CTYJ07 11501580 IC50 = 24000 nM T37848 C6ZN1O 11502217 IC50 > 10000 nM T37848 C3ME1U 11502912 IC50 = 17000 nM T37848 C2FWS0 11504172 IC50 = 5600 nM T37848 CFSH67 11504490 IC50 > 10000 nM T37848 C97WGN 11505187 IC50 = 5600 nM T37848 CLPO39 11508317 IC50 > 10000 nM T37848 CQ6IU7 11509269 IC50 > 10000 nM T37848 CJP81E 11510084 IC50 = 3400 nM T37848 CE76UG 11510297 IC50 = 29000 nM T37848 CRV87M 11510548 IC50 = 160 nM T37848 C8M0VI 11511019 IC50 = 7000 nM T37848 C2T8YD 11511361 IC50 > 10000 nM T37848 CP8B7T 11511719 IC50 = 1800 nM T37848 C29SZQ 11512193 IC50 = 1400 nM T37848 CDQ18N 11515125 IC50 > 10000 nM T37848 CP9RB7 11515387 IC50 > 10000 nM T37848 C0SN2O 11515728 IC50 > 10000 nM T37848 COTH53 11516139 IC50 = 84000 nM T37848 CVNP35 11517292 IC50 > 10000 nM T37848 CGA5W8 11519085 IC50 = 9000 nM T37848 C0QK6P 11519336 IC50 > 10000 nM T37848 CX4MA8 11519486 IC50 = 10000 nM T37848 CY47AQ 11519784 IC50 > 10000 nM T37848 CVO7T9 11522969 IC50 > 10000 nM T37848 CVPX30 11523521 IC50 = 38000 nM T37848 C2D8PW 11524511 IC50 = 25700 nM T37848 C4GLJ5 11524843 IC50 > 10000 nM T37848 CT1WQ3 11525337 IC50 = 5700 nM T37848 CGC86O 11525338 IC50 = 2600 nM T37848 C8H9KG 11526278 IC50 = 7000 nM T37848 C18QBV 11526524 IC50 = 2200 nM T37848 CMC5B1 11526626 IC50 > 10000 nM T37848 CSV8N7 11526667 IC50 = 1000 nM T37848 CR71GB 11526691 IC50 = 1500 nM T37848 C7HNP0 11526745 IC50 = 1200 nM T37848 C0BF5R 11527661 IC50 > 25000 nM T37848 C75FPD 11529874 IC50 > 3000 nM T37848 CRJC25 11530171 IC50 > 10000 nM T37848 C0BC6Y 11530223 IC50 > 10000 nM T37848 C4W2IN 11533195 IC50 = 20600 nM T37848 C4Q8VK 11533340 IC50 > 10000 nM T37848 CFU5V9 11533398 IC50 > 10000 nM T37848 CI8PW4 11533783 IC50 > 40000 nM T37848 CI82YU 11534139 IC50 = 2 nM T37848 CR92GA 11537005 IC50 = 850 nM T37848 CQZ82F 11539239 IC50 > 10000 nM T37848 CF2OM8 11539410 IC50 > 50000 nM T37848 CZ68TF 11540571 IC50 = 5200 nM T37848 CVX6L8 11541073 IC50 > 10000 nM T37848 C8P5GF 11541506 IC50 > 10000 nM T37848 C3VP9T 11544537 IC50 > 10000 nM T37848 C8P4XE 11546950 IC50 = 2600 nM T37848 C82BTJ 11547150 IC50 = 14900 nM T37848 C7IOJ0 11548023 IC50 = 2500 nM T37848 CE59MD 11548497 IC50 = 7600 nM T37848 C34JAV 11551351 IC50 > 10000 nM T37848 CN4MY1 11553111 IC50 = 36600 nM T37848 CUAI98 11555639 IC50 > 30 nM T37848 C86MYU 11559484 IC50 > 50000 nM T37848 CJN1E0 11561190 IC50 = 700 nM T37848 C17MUY 11561279 IC50 = 9300 nM T37848 CACS26 11561968 IC50 = 20800 nM T37848 CD9SM0 11562361 IC50 = 2300 nM T37848 C3KWU8 11562728 IC50 > 40000 nM T37848 C7B4YX 11563243 IC50 > 10000 nM T37848 C84NIF 11566130 IC50 > 10000 nM T37848 CDFU34 11566489 IC50 > 10000 nM T37848 CZ79RA 11566856 IC50 = 76000 nM T37848 CB59HM 11570626 IC50 = 60000 nM T37848 C4IX6W 11573549 IC50 > 10000 nM T37848 CP68BA 11575755 IC50 = 1000 nM T37848 CTVX46 11576269 IC50 = 6400 nM T37848 CF0UV9 11576464 IC50 = 30 nM T37848 CR75FZ 11577204 IC50 = 9300 nM T37848 CSJ5E1 11577280 IC50 = 4800 nM T37848 CXP2M0 11580426 IC50 > 10000 nM T37848 CW7G3X 11580427 IC50 > 10000 nM T37848 CVX6K7 11580514 IC50 > 10000 nM T37848 C3YXZ7 11582291 IC50 = 27000 nM T37848 CKW1Z2 11582790 IC50 = 344 nM T37848 CO9KP5 11583459 IC50 = 17000 nM T37848 CXJ8W9 11584004 IC50 > 10000 nM T37848 C4PTW2 11584329 IC50 > 40000 nM T37848 CFZ1Q5 11584681 IC50 = 29000 nM T37848 CFU15B 11588489 IC50 = 32000 nM T37848 C2H7WN 11590652 IC50 = 580 nM T37848 C1HG4A 11591164 IC50 = 22000 nM T37848 CWAZ43 11591353 IC50 = 400 nM T37848 C12PEW 11592380 IC50 = 5100 nM T37848 C2Q9YI 11596174 IC50 > 50000 nM T37848 C0Q9NP 11597977 IC50 = 9000 nM T37848 CHU90R 11598626 IC50 > 8000 nM T37848 C89AHL 11599077 IC50 = 1200 nM T37848 C28POG 11599126 IC50 = 3.2 nM T37848 CP56DO 11599295 IC50 > 10000 nM T37848 CR37EA 11602469 IC50 = 74000 nM T37848 C4ALS8 11602549 IC50 = 59000 nM T37848 C15TEH 11604449 IC50 > 10000 nM T37848 C0N5DY 11604763 IC50 = 1000 nM T37848 CYEN01 11605242 IC50 = 3400 nM T37848 CPH40V 11607042 IC50 > 30000 nM T37848 CH7P9Z 11608743 IC50 > 30000 nM T37848 C2M8HZ 11610353 IC50 > 50000 nM T37848 C42UWG 11610553 IC50 > 10000 nM T37848 CKXH63 11610910 IC50 > 12000 nM T37848 CM7LS0 11612187 IC50 = 5500 nM T37848 C1SL7N 11612461 IC50 = 2100 nM T37848 C6LUG4 11612700 IC50 = 6100 nM T37848 CAOU14 11613185 IC50 = 1.4 nM T37848 CL5OY4 11613524 IC50 = 300 nM T37848 C5JZ6R 11615459 IC50 > 40000 nM T37848 C9UI2V 11617038 IC50 = 26000 nM T37848 CW0ZM6 11619260 IC50 > 50000 nM T37848 CCYV36 11620477 IC50 > 40000 nM T37848 C79OMR 11623756 IC50 > 10000 nM T37848 CSB9O5 11623845 IC50 > 10000 nM T37848 CGX96V 11626927 IC50 < 50118.72 nM T37848 C3CP2G 11627368 IC50 = 1000 nM T37848 C7CG3P 11627369 IC50 = 1500 nM T37848 C3I6YE 11627465 IC50 = 13.8 nM T37848 C7H0RD 11628240 IC50 > 30 nM T37848 C9L5VD 11631813 IC50 > 50000 nM T37848 CQ2ZX6 11632274 IC50 = 2000 nM T37848 CM1DR9 11632375 IC50 = 1000 nM T37848 CN4R5G 11632540 IC50 = 3400 nM T37848 C7OF9S 11633939 IC50 = 4 nM T37848 CYL45U 11634544 IC50 = 3800 nM T37848 CDE1G8 11635187 IC50 = 40 nM T37848 CUN3R9 11635332 IC50 = 2020 nM T37848 CSKI72 11635565 IC50 = 2000 nM T37848 C23XSL 11638166 IC50 = 2800 nM T37848 CCP69D 11638499 IC50 > 9000 nM T37848 CRT09O 11638500 IC50 > 10000 nM T37848 C8C3PR 11639062 IC50 = 2500 nM T37848 COF14U 11641059 IC50 = 11900 nM T37848 CT4BE7 11641076 IC50 = 7900 nM T37848 CJS28X 11641672 IC50 = 2700 nM T37848 CQRB62 11641686 IC50 = 2500 nM T37848 CTXG50 11642625 IC50 = 1700 nM T37848 CBI47S 11645773 IC50 = 59000 nM T37848 C8GS9Z 11646163 IC50 > 50000 nM T37848 C6Y4HR 11647548 IC50 > 30000 nM T37848 CU8SI9 11649179 IC50 = 5000 nM T37848 CMB6F9 11653874 IC50 > 50000 nM T37848 CB7P8J 11655677 IC50 = 30000 nM T37848 CX7FR8 11655728 IC50 > 9000 nM T37848 CM2T8F 11656187 IC50 = 5500 nM T37848 CH3N1I 11659592 IC50 = 4000 nM T37848 CF92SM 11659664 IC50 = 17900 nM T37848 CDOZ32 11661172 IC50 = 100 nM T37848 CG54AP 11661821 IC50 = 10000 nM T37848 C3E0TV 11663187 IC50 = 4300 nM T37848 CO15KF 11664409 IC50 = 6700 nM T37848 C51UDK 11667741 IC50 > 10000 nM T37848 CXJ17M 11669364 IC50 = 50000 nM T37848 CS4R8Z 11670378 IC50 > 20000 nM T37848 CIUJ01 11670392 IC50 = 5000 nM T37848 C0V7SU 11675388 IC50 > 10000 nM T37848 C7JVX2 11681378 IC50 > 10000 nM T37848 C6M4TY 11681610 IC50 > 10000 nM T37848 C72BNQ 11682521 IC50 = 10000 nM T37848 CRF5P4 11685733 IC50 > 10000 nM T37848 CY36RI 11688223 IC50 > 10000 nM T37848 CW4U3H 11688520 IC50 > 10000 nM T37848 C2K9XG 11688776 IC50 = 10000 nM T37848 C3WBU8 11689242 IC50 = 48000 nM T37848 CM8R9J 11690073 IC50 = 260 nM T37848 CU0E8O 11690457 IC50 = 8300 nM T37848 C1OI3P 11690914 IC50 = 15000 nM T37848 C3YKD0 11691434 IC50 = 12600 nM T37848 C7Z0SX 11695591 IC50 > 10000 nM T37848 C9CM2R 11695689 IC50 > 50000 nM T37848 CP3G0Q 11695811 IC50 > 10000 nM T37848 COH3C4 11697546 IC50 = 350 nM T37848 CVL10S 11698924 IC50 = 1900 nM T37848 C5ECV1 11699447 IC50 > 35000 nM T37848 C4DJ1V 11699804 IC50 > 10000 nM T37848 CBDC74 11702114 IC50 > 10000 nM T37848 CQ5P2F 11702115 IC50 > 10000 nM T37848 CXFK83 11702578 IC50 > 10000 nM T37848 CU6D3X 11703421 IC50 = 4000 nM T37848 CO3U4B 11705008 IC50 = 300 nM T37848 CB0AP2 11705863 IC50 = 19600 nM T37848 C04VLB 11706579 IC50 > 10000 nM T37848 CL4DS1 11709762 IC50 > 10000 nM T37848 CK4I6J 11710700 IC50 = 1000 nM T37848 C5FZ1J 11710873 IC50 = 35000 nM T37848 C70LWD 11712638 IC50 = 17500 nM T37848 CHK5I2 11712756 IC50 = 5000 nM T37848 C6PFT9 11713201 IC50 = 0.8 nM T37848 CN5UX7 11713409 IC50 = 25000 nM T37848 CL5S9K 11719046 IC50 = 2300 nM T37848 C07CUH 11719337 IC50 = 3700 nM T37848 CZY05V 11719421 IC50 = 42000 nM T37848 CD9A0J 11720104 IC50 > 10000 nM T37848 CX9VH0 11720815 IC50 > 10000 nM T37848 C0Z5JS 11740023 IC50 = 18000 nM T37848 CI1P7M 11750760 IC50 = 640 nM T37848 CJXT34 11751643 IC50 = 210 nM T37848 CG0YB2 11751828 IC50 > 10000 nM T37848 CVSO90 11753013 IC50 = 6100 nM T37848 C58DMZ 11757696 IC50 = 12000 nM T37848 CNPX34 11757854 IC50 = 68 nM T37848 C8D7BS 11771234 IC50 = 3604 nM T37848 CB36OJ 11771503 IC50 > 40000 nM T37848 C6TS4D 11773824 IC50 = 1488 nM T37848 C9X6DU 11774980 IC50 = 12580 nM T37848 COI0P1 11774981 IC50 = 200 nM T37848 CLR59J 11775287 IC50 = 260 nM T37848 C6A1LM 11786814 IC50 > 500000 nM T37848 CN8CP5 11817019 IC50 = 29300 nM T37848 CS7W2V 11848793 IC50 > 30000 nM T37848 CQ26XH 11851431 IC50 = 60 nM T37848 C42BOS 11854299 IC50 = 1000 nM T37848 C2FN7G 11854301 IC50 = 1000 nM T37848 CI6JQ5 11855008 IC50 = 139000 nM T37848 CL1FX0 11947758 IC50 > 30000 nM T37848 CT0H7I 11949628 IC50 < 400 nM T37848 CPT14W 11962165 IC50 = 25000 nM T37848 CK2EZ6 11962967 IC50 >= 100000 nM T37848 CH26TZ 11963255 IC50 > 100000 nM T37848 C8P9GD 11966041 IC50 > 10000 nM T37848 CYEN98 11977494 IC50 = 66200 nM T37848 CN5W3V 11978858 IC50 = 42600 nM T37848 CW8T4V 11978859 IC50 = 41700 nM T37848 CW69VS 11993730 IC50 = 13000 nM T37848 CM07WK 11993787 IC50 > 2000 nM T37848 C1T8XZ 11993865 Ki > 400000 nM T37848 CBZ83S 11993868 Ki > 400000 nM T37848 C7A1EZ 11993870 Ki > 400000 nM T37848 C4XP2N 11993872 Ki = 1500 nM T37848 CWT0S3 11993875 Ki = 95500 nM T37848 CR4YS2 11996303 IC50 > 10000 nM T37848 C7D1AY 11996304 IC50 > 10000 nM T37848 C1A2IB 12001199 IC50 > 100000 nM T37848 CK90JR 12001280 IC50 = 5600 nM T37848 C2JP6D 12001701 IC50 > 7000 nM T37848 CV1IS7 12001783 IC50 = 4800 nM T37848 C2HV4P 12001784 IC50 = 3200 nM T37848 C2QAW5 12001786 IC50 = 3100 nM T37848 CQKJ25 12001869 IC50 = 4000 nM T37848 CF0C8W 12001871 IC50 = 5100 nM T37848 CHE5V2 12001872 IC50 = 16000 nM T37848 C2F1JZ 12001873 IC50 = 15000 nM T37848 CK7CQ0 12001952 IC50 = 2800 nM T37848 CM68CQ 12001953 IC50 = 15000 nM T37848 C17AVT 12001954 IC50 = 2400 nM T37848 CS5BA8 12001955 IC50 = 7300 nM T37848 CL6OY0 12001956 IC50 = 14000 nM T37848 C0EPD3 12039019 IC50 = 1600 nM T37848 C13GAW 12043371 IC50 = 4900 nM T37848 CZJ0B5 12043372 IC50 = 3700 nM T37848 C85ZFQ 12043374 IC50 = 7600 nM T37848 CF28CA 12074093 IC50 > 10000 nM T37848 CJY17R 12074102 IC50 > 10000 nM T37848 CJV5G1 12074103 IC50 = 5400 nM T37848 CNTU10 12082365 IC50 = 810 nM T37848 C9RX1L 12108566 IC50 = 40 nM T37848 CVIZ19 12112546 IC50 = 600 nM T37848 C3L8ZX 12312690 IC50 > 100000 nM T37848 CW7EC6 12854713 IC50 = 897 nM T37848 CO3HN1 13163256 IC50 > 100000 nM T37848 C7I9PF 13557523 Ki > 400000 nM T37848 C0FY4P 13615899 IC50 = 10600 nM T37848 C1G0EZ 13957609 IC50 = 520 nM T37848 C7EF6T 14179008 IC50 = 4 nM T37848 C9JY7V 14179009 IC50 = 17 nM T37848 C2LNX9 14179010 IC50 = 16 nM T37848 CEPW59 14179013 IC50 = 4 nM T37848 CIF90V 14434140 IC50 = 28000 nM T37848 CXS7Y5 14825858 IC50 = 31600 nM T37848 CR54KX 14861225 IC50 = 59000 nM T37848 C9VYL5 15172937 IC50 = 74000 nM T37848 C3YRU7 15295578 IC50 = 1300 nM T37848 C7X3CQ 15604497 IC50 = 10000 nM T37848 CXF80W 15604512 IC50 = 41000 nM T37848 CT4RL1 15778480 IC50 = 27000 nM T37848 CBE59I 15940927 IC50 = 30300 nM T37848 C08NEU 15945881 IC50 > 10000 nM T37848 CO7YL9 15947487 IC50 > 30000 nM T37848 C79VQK 15950271 IC50 > 10000 nM T37848 CU4P5X 15950383 IC50 = 1300 nM T37848 C16XRI 15950384 IC50 = 770 nM T37848 CUMR27 15950385 IC50 = 2500 nM T37848 C69RAY 15950386 IC50 = 1400 nM T37848 CM63YP 15950387 IC50 = 730 nM T37848 CH8F7W 15950388 IC50 = 670 nM T37848 C0L4SH 15950456 IC50 > 40000 nM T37848 C8FU1V 15950462 IC50 > 40000 nM T37848 C9KJ6D 15950538 IC50 = 17000 nM T37848 C4S7AB 15950540 IC50 > 40000 nM T37848 C3U1VO 15950542 IC50 > 40000 nM T37848 CKX8M6 15950615 IC50 = 22000 nM T37848 C3BI9R 15951010 IC50 > 10000 nM T37848 CWH1A8 15951076 IC50 > 10000 nM T37848 C2ZYA6 15951338 IC50 = 57300 nM T37848 C1Q8IV 15951410 IC50 = 23100 nM T37848 CC0M2X 15951427 IC50 = 1200 nM T37848 CF3PX0 15951428 IC50 = 2800 nM T37848 CWTX01 15951429 IC50 = 270 nM T37848 C3LQD9 15951431 IC50 = 390 nM T37848 CD59BN 15954476 IC50 = 50 nM T37848 CUI7P4 15955613 IC50 < 1000 nM T37848 C8QH9A 15958769 IC50 = 1000 nM T37848 C3W8ZL 15981007 IC50 > 50000 nM T37848 CW6S0H 15981486 IC50 = 1600 nM T37848 C7SN1C 15983053 IC50 = 3300 nM T37848 CS97JR 15983175 IC50 > 20000 nM T37848 C0O5BA 15983546 IC50 > 50000 nM T37848 C83NXU 15983672 IC50 = 4500 nM T37848 C2D1KP 15983982 IC50 = 330 nM T37848 CU2LO6 15984134 IC50 = 69000 nM T37848 C46QET 15984241 IC50 = 18000 nM T37848 C2VR7O 15984242 IC50 = 8700 nM T37848 CMX86T 15984318 IC50 = 4700 nM T37848 C5YH9J 15984938 IC50 = 14000 nM T37848 C5PCN0 15984939 IC50 = 58000 nM T37848 CQJ7Y2 15985912 IC50 = 3981.07 nM T37848 CPR25X 15986917 IC50 = 100000 nM T37848 C5KW3L 15987108 IC50 > 100000 nM T37848 CCL59Z 16007088 IC50 > 10000 nM T37848 C08CSK 16007091 IC50 > 18000 nM T37848 CG5A7W 16013152 IC50 = 1700 nM T37848 CBMF65 16013184 IC50 = 5700 nM T37848 C6V4TG 16013186 IC50 = 5300 nM T37848 C20CRP 16040587 IC50 = 1400 nM T37848 C8ZP3G 16041292 IC50 = 46000 nM T37848 CDU1L0 16041411 IC50 > 60000 nM T37848 CI6L0N 16042459 IC50 = 400 nM T37848 CMZU26 16043268 IC50 = 1140 nM T37848 C29KFG 16045493 IC50 = 4400 nM T37848 CU27FI 16049886 IC50 > 25000 nM T37848 CZC7L2 16049887 IC50 > 25000 nM T37848 CQ9U1Y 16051921 IC50 = 28000 nM T37848 CE43QM 16064288 IC50 = 34000 nM T37848 CELY15 16064449 IC50 > 40000 nM T37848 C8UOX0 16064748 IC50 = 7100 nM T37848 CFKE48 16064750 IC50 = 10000 nM T37848 CC7QD3 16064891 IC50 = 26000 nM T37848 CLG6R7 16064892 IC50 = 3300 nM T37848 C0C2QW 16064893 IC50 = 3400 nM T37848 C30UFT 16066811 IC50 > 50000 nM T37848 CFK8J5 16068056 IC50 = 2280 nM T37848 CQRU95 16070337 IC50 = 5000 nM T37848 C8E6CH 16070448 IC50 = 1000 nM T37848 CTIQ90 16071896 IC50 = 5000 nM T37848 CX2GC6 16071897 IC50 = 1000 nM T37848 CL4ON2 16072021 IC50 = 25000 nM T37848 CJU50N 16072099 IC50 = 1620 nM T37848 CIV72W 16086657 IC50 > 10000 nM T37848 C8D0KF 16099905 IC50 = 7000 nM T37848 C2FXW0 16099923 IC50 = 55000 nM T37848 C37LJV 16102853 IC50 > 50000 nM T37848 CEF3A0 16102867 IC50 = 1000 nM T37848 C91AZO 16102868 IC50 = 7200 nM T37848 CX5KI3 16105788 IC50 > 10000 nM T37848 CC24LB 16110489 IC50 > 10000 nM T37848 CJO58L 16116998 IC50 > 25000 nM T37848 C9HI7G 16118895 IC50 = 7700 nM T37848 CT3YW2 16118896 IC50 > 50000 nM T37848 CF7M3V 16118899 IC50 = 6100 nM T37848 C8ZEG9 16118900 IC50 = 4800 nM T37848 CHR8G4 16122633 IC50 = 10000 nM T37848 C0S1VK 16122818 IC50 > 40000 nM T37848 CFYL31 16122898 IC50 > 50000 nM T37848 C9G8TZ 16124598 IC50 = 100000 nM T37848 C0J6CH 16125372 IC50 = 91900 nM T37848 CMN0P3 16125681 IC50 > 100000 nM T37848 C4BYI2 16125682 IC50 > 100000 nM T37848 C8FLH6 16202152 IC50 = 10000 nM T37848 CWJZ50 16223655 IC50 = 1.4 nM T37848 CDG38L 16223656 IC50 > 10 nM T37848 C3O7HD 16223851 IC50 = 4.7 nM T37848 C0D9KR 16223854 IC50 = 15.1 nM T37848 C5L1QM 16224456 IC50 > 50 nM T37848 CU06JN 16225483 IC50 = 270 nM T37848 C9CL7E 16249526 Ki = 540 nM T37848 CTH6W4 16292141 IC50 > 25000 nM T37848 CQ3HO2 16309462 IC50 > 20000 nM T37848 C2V9PA 16432893 Ki = 11900 nM T37848 CIH5F7 16432896 Ki = 3900 nM T37848 CBM6Y7 16432965 Ki = 540 nM T37848 C07CYO 16432973 Ki = 700 nM T37848 CVJ4O1 16654686 Ki = 76000 nM T37848 C4QU0M 16654984 IC50 > 6000 nM T37848 CY6D1F 16656782 IC50 = 1900 nM T37848 C6P4BX 16656803 IC50 > 25000 nM T37848 CFW43X 16658022 IC50 = 500 nM T37848 C6H5VO 16658023 IC50 = 250 nM T37848 CC9W4S 16658024 IC50 = 250 nM T37848 CR51WX 16658101 IC50 = 80 nM T37848 CMLR19 16658102 IC50 = 250 nM T37848 CXN32U 16658103 IC50 = 200 nM T37848 C2XP7B 16658104 IC50 = 250 nM T37848 CD6L7Z 16658105 IC50 = 500 nM T37848 C7X0TS 16659334 IC50 > 30000 nM T37848 C9M0IS 16662085 IC50 = 1000 nM T37848 C5AB3F 16662086 IC50 = 1000 nM T37848 CRL96A 16662087 IC50 = 4000 nM T37848 C4L1FE 16662089 IC50 = 8000 nM T37848 CG9VH4 16662090 IC50 = 3500 nM T37848 CYJS23 16662091 IC50 = 3000 nM T37848 CU0V6D 16662092 IC50 = 10000 nM T37848 C2AL3D 16662093 IC50 = 10000 nM T37848 CSW16Z 16662094 IC50 = 10000 nM T37848 CR8I4H 16662096 IC50 = 4000 nM T37848 C5FH6G 16662098 IC50 = 470 nM T37848 CA2OZ7 16662100 IC50 = 530 nM T37848 C2UTD6 16662102 IC50 = 250 nM T37848 CZ9I1L 16662104 IC50 = 7000 nM T37848 CUI6P9 16662106 IC50 = 10000 nM T37848 C8CIQ4 16662108 IC50 = 410 nM T37848 CS08VM 16662110 IC50 > 10000 nM T37848 C6Y1GR 16662112 IC50 = 450 nM T37848 C5O6UF 16662114 IC50 = 1000 nM T37848 C9D6UT 16662116 IC50 = 170 nM T37848 CQ8U7P 16662118 IC50 = 490 nM T37848 CXL4Q3 16663122 IC50 = 58100 nM T37848 CK4FJ8 16664733 IC50 > 20000 nM T37848 C1UY8J 16666386 IC50 = 10000 nM T37848 CH0Q9T 16678616 IC50 > 50000 nM T37848 C4FUO7 16678620 IC50 = 6000 nM T37848 CDY08B 16678725 IC50 > 50000 nM T37848 C1N8IL 16679518 IC50 > 50000 nM T37848 C0CF9G 16679612 IC50 > 50000 nM T37848 C8X6SN 16679614 IC50 = 26000 nM T37848 CH8A2G 16679616 IC50 > 50000 nM T37848 CBE9O8 16679617 IC50 > 50000 nM T37848 CQF5Y7 16679701 IC50 > 50000 nM T37848 CSK8N5 16679707 IC50 > 50000 nM T37848 CI1J6W 16681732 IC50 = 3500 nM T37848 CK9IU2 16718491 IC50 = 8200 nM T37848 CAPU50 16719554 IC50 = 10000 nM T37848 CN95DG 16719649 IC50 > 100000 nM T37848 C92NRU 16727109 IC50 > 40000 nM T37848 CG04RZ 16727123 IC50 = 700 nM T37848 COJU37 16727124 IC50 > 50000 nM T37848 CAX2B7 16728787 IC50 > 30000 nM T37848 C0H8UN 16730109 IC50 > 40000 nM T37848 C9BC0L 16732000 IC50 > 40000 nM T37848 CHU72I 16738321 IC50 = 360 nM T37848 CBR95H 16739953 IC50 = 3600 nM T37848 CLY57P 16744597 IC50 > 40000 nM T37848 CA68OS 16744599 IC50 = 40000 nM T37848 CUI0X4 16744748 IC50 > 40000 nM T37848 CM3OV0 16745085 IC50 = 13000 nM T37848 C94MKR 16745086 IC50 = 32000 nM T37848 C5GY6N 16745241 IC50 = 24000 nM T37848 CW85LQ 16745311 IC50 = 2480 nM T37848 CC4L1M 16747701 IC50 > 22000 nM T37848 CW2SY5 16750291 IC50 > 10000 nM T37848 CIX7U2 16750304 IC50 > 10000 nM T37848 C4AZ3J 16752689 IC50 = 200 nM T37848 C5DKZ8 16956771 IC50 > 11000 nM T37848 CU42ZC 17244953 IC50 = 10000 nM T37848 C8D4PX 17408359 IC50 = 14000 nM T37848 C8O3JV 17720407 Ki = 14500 nM T37848 C9C5TV 17751819 IC50 > 50000 nM T37848 C8TKD5 17754437 IC50 > 100000 nM T37848 CAJ0S2 17754557 EC50 > 50000 nM T37848 C5XFD3 17757326 IC50 = 3600 nM T37848 CIE58R 17758239 IC50 = 16000 nM T37848 CWH37T 17758574 IC50 = 15000 nM T37848 C57NRL 17759787 IC50 = 18000 nM T37848 CT5L0Q 17955460 IC50 > 10000 nM T37848 CC9BE5 17963726 IC50 < 1000 nM T37848 C87WIK 18104758 IC50 > 50000 nM T37848 CF9TW8 18414685 IC50 = 9000 nM T37848 CG93TR 18440026 IC50 = 24000 nM T37848 C0YIF1 18440270 IC50 = 600 nM T37848 C1QM2U 18440271 IC50 = 410 nM T37848 CWQD08 18548739 IC50 < 100 nM T37848 CK2AJ8 18668528 IC50 = 2400 nM T37848 CI3HL4 18668538 IC50 > 10000 nM T37848 CCWH59 18668580 IC50 > 10000 nM T37848 CW8PF5 18668583 IC50 = 1000 nM T37848 C6ADH5 18668593 IC50 = 7100 nM T37848 C4-JAN-02 18668607 IC50 = 5500 nM T37848 C9V4BO 18668614 IC50 = 8100 nM T37848 CY1HK4 18668617 IC50 > 10000 nM T37848 CTA76E 18769059 IC50 = 3600 nM T37848 C7UKI6 18769065 IC50 > 10000 nM T37848 C0LCW3 18769074 IC50 > 10000 nM T37848 C8QA0F 18769127 IC50 = 3700 nM T37848 C2HFY3 19553304 IC50 = 11800 nM T37848 CKH72O 20115797 IC50 > 50000 nM T37848 C1F3NK 20725561 IC50 > 10000 nM T37848 CR1K3H 20763282 IC50 = 51000 nM T37848 C8X0RI 20763372 IC50 > 100000 nM T37848 C8OHP4 20763385 IC50 > 100000 nM T37848 C6POY9 20763386 IC50 = 65000 nM T37848 CZBJ32 20763421 IC50 = 94000 nM T37848 C7OMR1 20763606 IC50 > 100000 nM T37848 C81JWV 20906619 IC50 = 8000 nM T37848 CW3VX1 21018389 IC50 = 160 nM T37848 C57CRP 21036878 IC50 = 13000 nM T37848 CQ91KY 21049437 IC50 = 400 nM T37848 CHC4Q3 21064283 IC50 = 24900 nM T37848 C1CA6D 21070989 IC50 > 10000 nM T37848 CZ1Q0N 21102224 IC50 < 1000 nM T37848 CY9B5M 21257907 IC50 = 2100 nM T37848 CO17PU 21635104 IC50 = 19952.62 nM T37848 CO6E2Z 21717336 IC50 = 5500 nM T37848 C7KIJ3 21717337 IC50 = 4700 nM T37848 CKV94G 21879620 IC50 < 1000 nM T37848 C2KMV5 21879624 IC50 > 10000 nM T37848 CW8M5K 21899433 IC50 = 100 nM T37848 CM1IF8 21914519 IC50 > 100000 nM T37848 CZF82E 21914667 IC50 > 63095.73 nM T37848 CB5M3Q 21936345 IC50 < 500 nM T37848 CK8X7S 21956341 IC50 = 16000 nM T37848 C3DT1N 22018410 IC50 = 1400 nM T37848 CXMA20 22018425 IC50 < 1000 nM T37848 C6CLB8 22224657 IC50 = 1 nM T37848 CZK6M0 22239024 IC50 = 3100 nM T37848 CO32YX 22254068 IC50 = 4100 nM T37848 C4YP8N 22431956 IC50 > 20000 nM T37848 CV8QK7 22448579 IC50 = 1 nM T37848 C9N5XW 22520172 IC50 > 20000 nM T37848 CT24BF 22664964 IC50 = 1400 nM T37848 C0F4YM 22737877 IC50 = 5700 nM T37848 CH3PO5 22966419 IC50 = 5000 nM T37848 C2BJY9 23395723 IC50 = 31000 nM T37848 CH3RP0 23395766 IC50 = 15000 nM T37848 C0G8KF 23395772 IC50 = 30000 nM T37848 CXP67J 23395785 IC50 = 19000 nM T37848 C32CYB 23395790 IC50 = 6000 nM T37848 C8A9OF 23395792 IC50 = 10000 nM T37848 CE1J3W 23395801 IC50 = 5000 nM T37848 CUXA85 23395806 IC50 = 2000 nM T37848 C01DHS 23395807 IC50 = 17000 nM T37848 CU2J0M 23395808 IC50 > 500 nM T37848 C3TVL7 23501721 IC50 > 7500 nM T37848 CF81SW 23582412 IC50 > 100000 nM T37848 C9K1DY 23583191 IC50 = 18000 nM T37848 CQSB59 23586140 IC50 = 455 nM T37848 CW2R4M 23624283 IC50 = 76000 nM T37848 CO1NA8 23624297 IC50 = 4770 nM T37848 CQ29HW 23626128 IC50 = 6800 nM T37848 C0HA4Y 23626131 IC50 > 20000 nM T37848 C3Z6LM 23626132 IC50 > 20000 nM T37848 C2EXB1 23626439 IC50 > 20000 nM T37848 C7EK4A 23626924 IC50 = 10700 nM T37848 CW6OB1 23627212 IC50 > 10000 nM T37848 C7HSL4 23628221 IC50 = 2800 nM T37848 CYRO10 23628222 IC50 = 8000 nM T37848 CWAT04 23630291 IC50 = 1200 nM T37848 CMQ6W7 23630305 IC50 = 500 nM T37848 CC29GD 23633277 IC50 = 1700 nM T37848 CU1LK3 23633350 IC50 <= 3000 nM T37848 CVF78O 23634281 IC50 <= 3000 nM T37848 C0RM6I 23635105 IC50 = 8300 nM T37848 CB45UM 23635106 IC50 = 9000 nM T37848 CFNQ06 23635107 IC50 = 6900 nM T37848 CPE8L0 23635108 IC50 = 6400 nM T37848 CDC19H 23635109 IC50 = 6800 nM T37848 CHU29W 23635235 IC50 = 9200 nM T37848 CWL5K4 23635236 IC50 = 6000 nM T37848 CVFQ41 23635237 IC50 = 10000 nM T37848 C9WSK4 23642165 IC50 = 5100 nM T37848 C9KA1C 23644725 IC50 = 18 nM T37848 C5L8SH 23644726 IC50 = 3790 nM T37848 CDL4G9 23645678 IC50 > 200000 nM T37848 CTB09J 23647311 IC50 = 2000 nM T37848 CJ6XT7 23647314 IC50 = 790 nM T37848 C1AQ9P 23647882 IC50 > 22000 nM T37848 CTJ2P1 23647883 IC50 > 30000 nM T37848 CU6E5F 23647884 IC50 = 3000 nM T37848 C6NS9I 23647885 IC50 > 30000 nM T37848 CD9IC3 23647886 IC50 = 860 nM T37848 CPX95O 23647887 IC50 = 460 nM T37848 CK9D8P 23647888 IC50 = 920 nM T37848 CX50BA 23647889 IC50 = 120 nM T37848 C37JMS 23647890 IC50 = 590 nM T37848 CJ97BQ 23647892 IC50 = 1900 nM T37848 CXP2G5 23647893 IC50 > 30000 nM T37848 C3JBX4 23647894 IC50 = 530 nM T37848 C71DGY 23647895 IC50 = 30000 nM T37848 C5LU8P 23647897 IC50 = 4790 nM T37848 C2YVQ3 23647898 IC50 = 1670 nM T37848 C4H5PR 23647899 IC50 = 160 nM T37848 CW6Y9I 23647900 IC50 > 30000 nM T37848 CMF8R6 23647901 IC50 = 2180 nM T37848 CR7CO9 23647902 IC50 = 670 nM T37848 CX37CO 23647903 IC50 > 30000 nM T37848 CMG8T2 23647904 IC50 = 270 nM T37848 C9H7NY 23647905 IC50 = 1060 nM T37848 C3MSV0 23647907 IC50 = 1700 nM T37848 C2Z0KQ 23647908 IC50 = 10000 nM T37848 CF9EK5 23647910 IC50 = 12000 nM T37848 CB1PL5 23647911 IC50 = 42 nM T37848 CQ9I4F 23647912 IC50 = 54 nM T37848 C9H0EC 23647913 IC50 = 10000 nM T37848 CN61YJ 23647914 IC50 = 15000 nM T37848 CZ0QF1 23648867 IC50 > 30000 nM T37848 CK76FP 23649427 IC50 > 100 nM T37848 CAUC58 23649669 IC50 > 100000 nM T37848 CCL15O 23652787 IC50 = 4610 nM T37848 CKW7V5 23653135 IC50 = 5540 nM T37848 CG39XH 23654666 IC50 > 100 nM T37848 C6VSO8 23657438 IC50 = 5000 nM T37848 CFMX27 23658550 IC50 = 130 nM T37848 C26ANU 23696680 IC50 = 35000 nM T37848 CASU54 23696973 IC50 >= 100000 nM T37848 CS5E6J 23729988 IC50 > 900000 nM T37848 CJYO24 24178214 IC50 = 67000 nM T37848 C8ONS6 24178219 IC50 = 97000 nM T37848 CO01RG 24178536 IC50 > 100000 nM T37848 C6FM9C 24180452 IC50 = 2200 nM T37848 CK2Q5J 24180592 IC50 > 10000 nM T37848 C0QI2D 24180593 IC50 = 16000 nM T37848 C7SMW5 24180646 IC50 = 4900 nM T37848 C9R1PK 24180717 IC50 > 20000 nM T37848 CN9S3A 24517908 IC50 = 1000 nM T37848 CZ03FI 24649020 IC50 > 50000 nM T37848 CUW7F4 24739481 IC50 = 1600 nM T37848 C2K1EL 24740535 IC50 = 1900 nM T37848 CD90WZ 24740655 IC50 = 6000 nM T37848 C2S3RO 24741625 IC50 = 170 nM T37848 C80ACG 24742640 IC50 = 5900 nM T37848 CQ35ZB 24743795 IC50 > 50000 nM T37848 C8RC9P 24744325 IC50 > 10000 nM T37848 CSG9V8 24749508 IC50 > 100000 nM T37848 C6JF2R 24753412 IC50 = 14000 nM T37848 C4CY3V 24753607 IC50 = 5600 nM T37848 CP1E4R 24753786 IC50 > 100000 nM T37848 COAY09 24753878 IC50 = 11000 nM T37848 CHU49V 24757938 IC50 > 50000 nM T37848 C25HKJ 24758044 IC50 > 40000 nM T37848 CJL67N 24759089 IC50 > 10000 nM T37848 C3OY6A 24759171 IC50 = 87 nM T37848 CET32I 24762429 IC50 > 100000 nM T37848 C1WHD0 24762502 IC50 > 100000 nM T37848 CK6NV1 24762503 IC50 > 100000 nM T37848 CSYQ45 24762504 IC50 > 100000 nM T37848 CR9ZI2 24764491 IC50 > 50000 nM T37848 CG23NJ 24768399 IC50 = 60 nM T37848 CSL71N 24768413 IC50 = 13000 nM T37848 C3P7IS 24768572 IC50 > 50000 nM T37848 C3AM6Z 24779751 IC50 = 400 nM T37848 C6ORA8 24783140 IC50 > 10000 nM T37848 CXSZ08 24783396 IC50 = 9300 nM T37848 CJ9Z1C 24796588 IC50 > 65000 nM T37848 CUM03S 24798754 IC50 > 50000 nM T37848 CV1JW8 24802616 IC50 = 32000 nM T37848 CR48VC 24809711 IC50 = 2000 nM T37848 CY8X0J 24811794 IC50 > 30000 nM T37848 C35JHQ 24812745 IC50 = 800 nM T37848 CK02ZF 24812771 IC50 > 50000 nM T37848 C6H2KZ 24817638 IC50 > 30000 nM T37848 C24UQW 24822428 IC50 = 13000 nM T37848 CROH43 24822429 IC50 = 100 nM T37848 C73LOX 24824080 IC50 = 160 nM T37848 CFI7E9 24824316 IC50 = 2000 nM T37848 CGDB50 24824447 IC50 = 40000 nM T37848 CLU56Y 24824450 IC50 > 50000 nM T37848 CF75DJ 24824494 IC50 = 510 nM T37848 C0CHG3 24824705 IC50 = 2000 nM T37848 C1B8TF 24825267 IC50 = 20000 nM T37848 C06COB 24825268 IC50 < 70 nM T37848 C47QTG 24825269 IC50 = 6700 nM T37848 CJ16YD 24825270 IC50 > 50000 nM T37848 CO1BL7 24825271 IC50 > 50000 nM T37848 CV0UB1 24825272 IC50 > 50000 nM T37848 CQN3Z7 24825710 IC50 > 40000 nM T37848 CN4Z2J 24825807 IC50 = 700 nM T37848 CM2Y0L 24827043 IC50 <= 1000 nM T37848 C6OJ5C 24827142 IC50 = 6000 nM T37848 CZI9P0 24829572 IC50 = 11400 nM T37848 C4T3UC 24829746 IC50 = 7400 nM T37848 C47LFZ 24830567 IC50 = 3800 nM T37848 C9E7AU 24830568 IC50 = 5000 nM T37848 CJ4K3P 24830569 IC50 = 7500 nM T37848 CKL92Z 24830570 IC50 = 5600 nM T37848 C2K1OE 24830571 IC50 > 30000 nM T37848 CP4KZ1 24830882 IC50 > 15000 nM T37848 C4J6AD 24831672 IC50 = 8300 nM T37848 C82YBD 24831841 IC50 = 3500 nM T37848 CTXJ06 24832008 IC50 = 1500 nM T37848 C75KOR 24832012 IC50 = 26000 nM T37848 CR7X1M 24856034 IC50 > 10000 nM T37848 CEW31B 24856362 IC50 > 100000 nM T37848 C61KPI 24856363 IC50 > 10000 nM T37848 CB4LY1 24857598 IC50 = 10000 nM T37848 CSR8J4 24857759 IC50 > 25000 nM T37848 CO73CZ 24862842 IC50 = 17000 nM T37848 C84JXU 24863323 IC50 = 23000 nM T37848 CUY1O2 24863332 IC50 = 30000 nM T37848 CV29XP 24863333 IC50 = 4000 nM T37848 CJIN21 24863334 IC50 = 11000 nM T37848 CM80JI 24863522 IC50 = 5000 nM T37848 CH6TG1 24864825 IC50 = 6400 nM T37848 CY2HJ0 24864993 IC50 = 8300 nM T37848 CEX30T 24865175 IC50 = 4800 nM T37848 C2X6ML 24867300 IC50 = 4 nM T37848 CM8BS1 24879232 IC50 > 5000 nM T37848 CK8XV4 24881399 IC50 = 3800 nM T37848 C4OE1F 24881534 IC50 = 300 nM T37848 CU29JQ 24882306 IC50 = 696 nM T37848 CX79IO 24882359 IC50 > 20000 nM T37848 CKRF92 24888487 IC50 = 13000 nM T37848 CU1G7V 24888656 IC50 = 3400 nM T37848 CF2H0Z 24888658 IC50 = 19000 nM T37848 CH9JZ4 24888820 IC50 = 7200 nM T37848 C45AQE 24889168 IC50 = 7200 nM T37848 C0Z2TG 24889346 IC50 = 2600 nM T37848 CDQ9I1 24889676 IC50 = 5100 nM T37848 CY8I0R 24889679 IC50 = 13000 nM T37848 C6NVP1 24889840 IC50 = 7200 nM T37848 CTE1I8 24889844 IC50 = 13000 nM T37848 CU18OW 24890344 IC50 = 1800 nM T37848 CUZ31Q 24890346 IC50 = 2100 nM T37848 C32TKP 24890348 IC50 = 1500 nM T37848 CBK4Z3 24890525 IC50 = 16000 nM T37848 CU4HV5 24890872 IC50 = 17000 nM T37848 CNQ6I4 24894028 IC50 > 20000 nM T37848 CE30NJ 24894058 IC50 > 40000 nM T37848 C1G6DM 24895969 IC50 < 1000 nM T37848 C59MRG 24896012 IC50 < 1000 nM T37848 C8FPH7 24896062 IC50 > 10000 nM T37848 C8C5JG 24896257 IC50 = 19500 nM T37848 CDI7N3 24897002 IC50 > 50000 nM T37848 C8GN9W 24899993 IC50 > 50000 nM T37848 CZSA05 24899995 IC50 > 50000 nM T37848 CIZ6O1 24900235 IC50 > 50000 nM T37848 C61ARF 24900236 IC50 > 50000 nM T37848 C7J4ZQ 24900259 IC50 > 40000 nM T37848 C0XW8P 24936070 IC50 = 11500 nM T37848 C83EUF 24937010 IC50 = 1500 nM T37848 C72LWC 24937637 IC50 = 1200 nM T37848 CC4K1P 24949545 IC50 = 1700 nM T37848 C17QKF 24949548 IC50 = 3900 nM T37848 CCA9G2 24949700 IC50 = 16000 nM T37848 CFU0T1 24949702 IC50 = 74000 nM T37848 CE79PI 24949704 IC50 = 1700 nM T37848 CI7NG8 24951587 IC50 > 8000 nM T37848 CLZ23U 24951610 IC50 > 30000 nM T37848 CNP3T1 24951733 IC50 > 50000 nM T37848 CEGV39 24951942 IC50 > 10000 nM T37848 C9EH3S 24951943 IC50 > 10000 nM T37848 CW9UN1 24951944 IC50 > 10000 nM T37848 CP98YL 24951946 IC50 > 10000 nM T37848 CCO20I 24953169 IC50 = 19600 nM T37848 CC0U6X 24953170 IC50 = 5600 nM T37848 CSEW45 24953255 IC50 = 150 nM T37848 CO41IK 24953519 IC50 = 1400 nM T37848 CJ43DG 24954671 IC50 = 3700 nM T37848 C0V8YL 24957182 IC50 = 2900 nM T37848 CCJ9G0 24958075 IC50 > 50000 nM T37848 C2UZ5G 24958816 IC50 > 10000 nM T37848 C8BEW0 24959168 IC50 > 50000 nM T37848 CNO0U1 24959169 IC50 > 10000 nM T37848 CBM71O 24959543 IC50 > 50000 nM T37848 C3VO7Q 24960588 IC50 = 4000 nM T37848 CZ89IP 24961687 IC50 = 2000 nM T37848 CW4X0E 24962988 IC50 > 3000 nM T37848 CB68JF 24963286 IC50 > 50000 nM T37848 C5EIW1 24965329 IC50 = 30500 nM T37848 C6U2AP 24965679 IC50 = 35970 nM T37848 CM6I1G 24967634 IC50 = 800 nM T37848 C0XS2D 24967990 IC50 = 3000 nM T37848 C71CNA 24967991 IC50 = 30000 nM T37848 CAN92Q 24968874 IC50 = 1400 nM T37848 CE95WV 24970356 IC50 = 220 nM T37848 CQ2Z7T 24985115 IC50 > 10000 nM T37848 CM7HQ5 24985395 IC50 > 20000 nM T37848 CEJ74C 24985745 IC50 > 20000 nM T37848 C27WVS 24986404 IC50 = 10000 nM T37848 C94AHE 24988956 IC50 = 62000 nM T37848 C0I5NG 24991884 IC50 = 79000 nM T37848 CL83OS 24992519 IC50 > 30000 nM T37848 CK0NZ8 24993163 IC50 > 10000 nM T37848 C8KIP6 24993178 IC50 > 30000 nM T37848 CD8U2B 24993500 IC50 > 30000 nM T37848 CCDF20 24994127 IC50 > 11000 nM T37848 CJM8R0 24996322 IC50 > 30000 nM T37848 C1T4WH 25003030 IC50 = 3300 nM T37848 CT64BR 25005273 IC50 = 1400 nM T37848 CX0O4A 25005628 IC50 > 50000 nM T37848 CR9LQ8 25005629 IC50 > 50000 nM T37848 C8ZQ3E 25005985 IC50 > 50000 nM T37848 C47CFM 25005986 IC50 > 50000 nM T37848 CKT5V7 25005987 IC50 > 50000 nM T37848 C5NF9P 25005988 IC50 = 9600 nM T37848 C2H8XF 25005989 IC50 = 25000 nM T37848 C1MWK0 25005990 IC50 > 50000 nM T37848 CX3I6O 25008509 IC50 = 9800 nM T37848 CBPY64 25008621 IC50 = 980 nM T37848 C0C3ZJ 25008854 IC50 > 10000 nM T37848 CX8N1E 25009027 IC50 = 800 nM T37848 C30HJO 25009028 IC50 = 4500 nM T37848 C3C6HW 25009031 IC50 = 3800 nM T37848 CZ6T5Q 25009937 IC50 > 29000 nM T37848 CU7G9E 25010550 IC50 < 10000 nM T37848 CBK82P 25011729 IC50 = 2600 nM T37848 C32AUW 25013308 IC50 > 10000 nM T37848 CP13LW 25016311 IC50 = 1600 nM T37848 C91QFN 25019282 IC50 = 37000 nM T37848 CMU30E 25022640 IC50 = 11000 nM T37848 CQ9LS6 25022704 IC50 > 3000 nM T37848 CF67EB 25023856 IC50 = 10000 nM T37848 C0L9PQ 25023857 IC50 < 10000 nM T37848 CA2T1X 25023858 IC50 < 10000 nM T37848 C7SKU1 25023859 IC50 < 10000 nM T37848 CA20NZ 25025581 IC50 > 9000 nM T37848 CPJD86 25025779 IC50 > 4000 nM T37848 CDX2C6 25025977 IC50 > 8000 nM T37848 C0LO9C 25028373 IC50 = 76000 nM T37848 CKLQ76 25028375 IC50 = 100000 nM T37848 CDKJ78 25033361 IC50 > 40000 nM T37848 C29WQM 25033651 IC50 = 3364 nM T37848 C1VPF8 25033652 IC50 = 13841 nM T37848 CDR34P 25033653 IC50 > 6947 nM T37848 CE0L8C 25033655 IC50 = 2394 nM T37848 C9Q8ZK 25033657 IC50 = 3643 nM T37848 CWIC10 25033659 IC50 = 357 nM T37848 C32QBZ 25033661 IC50 = 1697 nM T37848 CAI47X 25033725 IC50 = 2173 nM T37848 C1XW6O 25033727 IC50 = 632 nM T37848 C23EWR 25033729 IC50 = 3291 nM T37848 CW5A1U 25033730 IC50 = 8757 nM T37848 CV49HP 25033731 IC50 = 15190 nM T37848 CJHY97 25033732 IC50 = 159 nM T37848 C86AIT 25033734 IC50 = 4199 nM T37848 CEJ89P 25033804 IC50 = 2114 nM T37848 C3UF1V 25033806 IC50 = 1093 nM T37848 CF46OB 25033808 IC50 = 2300 nM T37848 CBI59C 25033810 IC50 = 3386 nM T37848 C0X8DC 25034109 IC50 = 84 nM T37848 CXDF80 25034348 IC50 = 9070 nM T37848 CZPW03 25034656 IC50 > 20000 nM T37848 C7KAR1 25034657 IC50 = 3231 nM T37848 CR3I9Y 25050394 EC50 = 1800 nM T37848 CVQS96 25052767 IC50 > 25000 nM T37848 CZO27W 25054032 IC50 = 8100 nM T37848 C7EQ5T 25054288 IC50 = 7700 nM T37848 CN2G3K 25054307 IC50 > 30000 nM T37848 C7EXD5 25054568 IC50 = 13500 nM T37848 C1PKF0 25056080 IC50 > 10000 nM T37848 CFHO90 25056112 IC50 = 5900 nM T37848 C6Z3CE 25057124 IC50 = 38000 nM T37848 CH6AU8 25057408 IC50 > 30000 nM T37848 C0B7RT 25057409 IC50 > 30000 nM T37848 C3AT0H 25057667 IC50 > 30000 nM T37848 CH7YC4 25057933 IC50 = 1700 nM T37848 CF7S1D 25064072 IC50 = 50000 nM T37848 C37HTN 25064073 IC50 = 4500 nM T37848 C9B0FR 25064510 IC50 = 14000 nM T37848 C6SZR4 25064730 IC50 = 41000 nM T37848 C6OCA7 25064916 IC50 > 10000 nM T37848 CID6R3 25065131 IC50 = 8900 nM T37848 CPT9X8 25066443 IC50 > 10000 nM T37848 CA76KJ 25067046 IC50 = 1400 nM T37848 CGMN97 25067404 IC50 > 30000 nM T37848 C7YRG0 25067560 IC50 = 100 nM T37848 CMH41V 25069448 IC50 = 40 nM T37848 CP3Y5K 25069603 IC50 > 20000 nM T37848 CM1WB9 25069914 IC50 > 20000 nM T37848 C8ANG7 25070193 IC50 = 4100 nM T37848 CBY3O2 25070582 IC50 > 30000 nM T37848 CM37LQ 25072736 IC50 = 100 nM T37848 C0UO6V 25073049 IC50 = 3400 nM T37848 C04QRE 25074004 IC50 = 2500 nM T37848 CBRM65 25074167 IC50 = 1070 nM T37848 C07GFA 25074313 IC50 > 20000 nM T37848 CLWN54 25074316 IC50 > 20000 nM T37848 C1AGW7 25093241 IC50 = 5300 nM T37848 CH90KV 25097876 IC50 > 10000 nM T37848 CAO38V 25098429 IC50 > 10000 nM T37848 CF7ON5 25099235 IC50 > 50000 nM T37848 CUYI02 25101821 IC50 > 10000 nM T37848 CSVP62 25106869 Ki = 18000 nM T37848 CLD7X0 25107258 IC50 = 2200 nM T37848 C4NE6H 25107259 IC50 = 1200 nM T37848 COT5G4 25107260 IC50 < 200 nM T37848 C0K9HA 25110600 IC50 > 14000 nM T37848 C4GSD8 25110702 IC50 = 3000 nM T37848 CR17NY 25110703 IC50 = 12000 nM T37848 C7I9MV 25110821 IC50 > 10000 nM T37848 CXBZ57 25118294 IC50 > 50000 nM T37848 CKRN07 25118654 IC50 > 50000 nM T37848 CJM41E 25119356 IC50 > 50000 nM T37848 C8HI9Y 25119357 IC50 > 50000 nM T37848 CGL63Q 25119716 IC50 > 50000 nM T37848 CG8D5U 25119991 IC50 = 1600 nM T37848 CQ8Y7T 25120419 IC50 > 50000 nM T37848 CXL3Q8 25121114 IC50 > 50000 nM T37848 C2S1LG 25121469 IC50 > 50000 nM T37848 C1RBQ7 25122183 IC50 > 50000 nM T37848 CYWO57 25122184 IC50 = 1400 nM T37848 CXO60C 25127299 IC50 = 1000 nM T37848 CNTF43 25127621 IC50 = 100 nM T37848 C4E0MJ 25127622 IC50 = 10000 nM T37848 CDO26T 25129042 IC50 > 31622.78 nM T37848 CP39AX 25132380 IC50 = 8000 nM T37848 CC5FH4 25132724 IC50 = 800 nM T37848 C3YH5W 25138072 IC50 = 43000 nM T37848 CMP7V1 25138073 IC50 > 20000 nM T37848 CLW7O5 25138074 IC50 = 8500 nM T37848 C7L6SP 25138075 IC50 = 740 nM T37848 C1PF5O 25138076 IC50 > 20000 nM T37848 CC4HW2 25138077 IC50 = 380 nM T37848 C9J1MQ 25138078 IC50 = 18000 nM T37848 C9LMW0 25138079 IC50 = 18000 nM T37848 C2QLK4 25138080 IC50 = 14000 nM T37848 CS89DE 25138081 IC50 > 20000 nM T37848 C5AJ0V 25138082 IC50 = 17000 nM T37848 CAL52B 25138083 IC50 = 16000 nM T37848 CZ41XS 25138084 IC50 = 20000 nM T37848 C9GZ6D 25138086 IC50 = 25000 nM T37848 C5A1FW 25138087 IC50 > 20000 nM T37848 CA01RE 25138089 IC50 > 20000 nM T37848 CC5O4P 25138090 IC50 > 20000 nM T37848 CQ30KW 25138091 IC50 = 11000 nM T37848 CCM9X1 25138092 IC50 > 20000 nM T37848 C9Z6UG 25138295 IC50 > 100000 nM T37848 CHS25Z 25141776 IC50 > 5000 nM T37848 CE93TF 25141777 IC50 > 5000 nM T37848 C1AIH7 25141896 IC50 > 5000 nM T37848 CZX08M 25142015 Ki = 33 nM T37848 CWF5Z3 25143506 IC50 > 30000 nM T37848 CFS3N9 25144422 IC50 > 20000 nM T37848 C78YWA 25145716 IC50 > 20000 nM T37848 C0VD1R 25154104 IC50 = 47000 nM T37848 CL9WT7 25154107 IC50 > 100000 nM T37848 C3O2FU 25154143 IC50 > 100000 nM T37848 CL1W5D 25154436 IC50 = 970 nM T37848 C67QXP 25154827 IC50 = 25200 nM T37848 C8AC0Y 25154864 IC50 = 1000 nM T37848 CWC26X 25156399 IC50 = 36000 nM T37848 CNOJ07 25156400 IC50 = 135000 nM T37848 C5Z1RT 25156669 IC50 = 29000 nM T37848 CQY6Z1 25156942 IC50 = 69000 nM T37848 CUE0Z5 25156943 IC50 = 11000 nM T37848 CQ6PI5 25156944 IC50 = 440 nM T37848 C5ZJX4 25156946 IC50 = 69000 nM T37848 CGH08V 25164128 IC50 = 4000 nM T37848 C3NVW5 25165471 IC50 > 15000 nM T37848 CF9KY4 25165474 IC50 > 30000 nM T37848 CH06WV 25168930 IC50 > 10000 nM T37848 C5TJD2 25172265 IC50 > 10000 nM T37848 CJMZ37 25174150 IC50 > 7500 nM T37848 C0XHA2 25180109 IC50 < 200000 nM T37848 C90UKD 25180304 IC50 = 12200 nM T37848 C6ZE9H 25180500 IC50 = 3800 nM T37848 CK6Z9J 25181419 IC50 = 64000 nM T37848 CL0Z1F 25181502 IC50 > 25000 nM T37848 CGE8V0 25181656 IC50 = 4600 nM T37848 CZUP40 25181801 IC50 = 13400 nM T37848 C5AKX1 25181802 IC50 = 5000 nM T37848 CF39AL 25182859 IC50 = 34000 nM T37848 C6EWF1 25183622 IC50 > 30000 nM T37848 C79LPB 25183668 IC50 = 4500 nM T37848 CHJY51 25183669 IC50 > 2000 nM T37848 C0Q8BN 25183817 IC50 > 20000 nM T37848 CF46YL 25183819 IC50 > 20000 nM T37848 C89CXW 25183820 IC50 > 20000 nM T37848 C5C7GH 25184832 IC50 > 10000 nM T37848 CSU0B5 25189891 IC50 > 15000 nM T37848 C04QGB 25190493 IC50 > 89000 nM T37848 CHN5O0 25190977 IC50 = 5000 nM T37848 CS3HT2 25191022 IC50 = 900 nM T37848 CV3TA6 25192021 IC50 > 7500 nM T37848 C9UL8Y 25192468 IC50 > 7500 nM T37848 C7A8UE 25192471 IC50 > 7500 nM T37848 CH3L6V 25192656 IC50 > 10000 nM T37848 C35EQD 25195745 IC50 = 37000 nM T37848 CVT64C 25196402 IC50 = 1800 nM T37848 C7BO9Q 25196404 IC50 = 700 nM T37848 C9TE8R 25196406 IC50 = 2700 nM T37848 C8CY6O 25205318 IC50 = 2000 nM T37848 CY1M9Q 25205319 IC50 = 1700 nM T37848 CEV2D7 25205475 IC50 = 940 nM T37848 C9S0ZW 25205477 IC50 = 5800 nM T37848 CLFM35 25206064 IC50 = 8600 nM T37848 C49KHR 25206116 IC50 = 570 nM T37848 CSGI69 25207352 IC50 = 40000 nM T37848 C37YTG 25210603 IC50 = 3000 nM T37848 CTQM87 25210756 IC50 > 100000 nM T37848 CE7BA0 25210873 IC50 = 4000 nM T37848 C2UQJ6 25211598 EC50 > 60000 nM T37848 CKI86X 25211805 EC50 > 60000 nM T37848 CHW2X0 25211910 EC50 > 100000 nM T37848 CXH7F8 25218692 IC50 > 20000 nM T37848 CDGF43 25218742 IC50 < 1000 nM T37848 CUN19O 25218744 IC50 = 4000 nM T37848 COWB90 25221040 IC50 = 3200 nM T37848 CC25TV 25222706 IC50 = 1300 nM T37848 CJ65AE 25226377 IC50 > 50000 nM T37848 C53PTZ 25256089 IC50 = 10000 nM T37848 CW9JM2 25256832 IC50 > 10000 nM T37848 C3GC7P 25256833 IC50 > 10000 nM T37848 CI8SQ7 25263541 IC50 = 15000 nM T37848 CTW7E8 25263542 IC50 > 20000 nM T37848 C03SUJ 25263865 IC50 = 13000 nM T37848 C6DX5M 25264621 IC50 = 660 nM T37848 C32USM 25264907 IC50 = 2800 nM T37848 CJ50IN 25265057 IC50 = 2200 nM T37848 C5E3ZH 25265089 IC50 > 100000 nM T37848 C20XDK 25265635 IC50 > 20000 nM T37848 CJ32HC 25265835 IC50 = 13600 nM T37848 C07DOP 26719840 IC50 = 8000 nM T37848 CI1G2C 26873419 IC50 = 3900 nM T37848 C9FCM8 29053150 IC50 = 1000000 nM T37848 C71FRE 35503002 IC50 > 33000 nM T37848 C0FA2X 40680501 IC50 = 50000 nM T37848 CE63OB 40700807 IC50 = 6000 nM T37848 CHW3D1 40700815 IC50 = 12500 nM T37848 CYL39Q 40924317 IC50 = 15000 nM T37848 CSU6D0 42171034 IC50 = 2900 nM T37848 CBH1P0 42210730 IC50 > 30000 nM T37848 CT0NF6 42415086 IC50 > 30000 nM T37848 C6AM3I 42598658 IC50 = 4000 nM T37848 CTQ8I9 42599146 IC50 = 1800 nM T37848 CKH3P1 42606928 IC50 > 40000 nM T37848 C30UMQ 42609861 IC50 = 31 nM T37848 C1YO7H 42618040 EC50 = 7000 nM T37848 CN34WV 42618054 EC50 = 7600 nM T37848 C0I4MK 42618066 EC50 = 4900 nM T37848 CGU3N8 42618068 EC50 = 1400 nM T37848 CY4LG8 42622934 IC50 > 75000 nM T37848 CJ8LY0 42626024 IC50 = 4700 nM T37848 CS04KE 42629368 IC50 > 100000 nM T37848 CYGN52 42629369 IC50 = 47000 nM T37848 CT97HP 42633319 IC50 = 1700 nM T37848 CGJ04I 42635527 IC50 = 19 nM T37848 CW4N5O 42635699 IC50 = 23 nM T37848 CH3MY1 42639933 IC50 > 27000 nM T37848 CVY8H2 42640092 IC50 > 27000 nM T37848 C9PL8Z 42641334 IC50 = 2600 nM T37848 C6MX0U 42641453 IC50 = 900 nM T37848 CFA3V2 42641819 IC50 = 260 nM T37848 C2D1MN 42642930 IC50 = 91 nM T37848 C4P1IM 42643589 IC50 < 10000 nM T37848 CX9SM6 42643591 IC50 < 10000 nM T37848 C96FIN 42644084 IC50 > 10000 nM T37848 C8BI5F 42644088 IC50 > 10000 nM T37848 CREJ31 42646199 IC50 > 100000 nM T37848 CKZ76R 42646202 IC50 > 10000 nM T37848 C81NVM 42646450 IC50 > 10000 nM T37848 CVBO78 42647178 IC50 < 10000 nM T37848 CZF5G9 42916879 IC50 > 10000 nM T37848 C5E6UL 43388611 IC50 = 5490 nM T37848 CS40ML 44123747 IC50 > 50000 nM T37848 C7VOU1 44126023 IC50 = 2400 nM T37848 CX7W2E 44132009 IC50 = 45000 nM T37848 CXS43I 44132271 IC50 = 320 nM T37848 CA0E4U 44132585 IC50 = 550 nM T37848 CA7HI4 44137226 IC50 > 10000 nM T37848 C5O1MR 44137674 IC50 > 10000 nM T37848 CG73ST 44138103 IC50 > 30000 nM T37848 CHR6C1 44141871 IC50 = 450000 nM T37848 C6QY9W 44143257 IC50 = 75000 nM T37848 CO2G0S 44155541 IC50 > 10000 nM T37848 CD4N7Z 44155649 IC50 > 10000 nM T37848 C65VWT 44155756 IC50 > 10000 nM T37848 CS5A1G 44157716 IC50 < 400 nM T37848 C3RKI7 44158698 IC50 > 50000 nM T37848 CO60AP 44159044 IC50 = 2400 nM T37848 C5G4LN 44159411 IC50 > 30000 nM T37848 CHI65U 44159530 IC50 = 18000 nM T37848 C9RC2Z 44159640 IC50 = 12000 nM T37848 C1C2DH 44159759 IC50 = 29000 nM T37848 CMNH53 44159772 IC50 = 21000 nM T37848 C5GYS4 44160248 IC50 > 50000 nM T37848 C38DTW 44160263 IC50 > 40000 nM T37848 CPF50A 44184875 IC50 > 24000 nM T37848 C2XE7Y 44189733 IC50 > 100000 nM T37848 CYJ7S2 44190263 IC50 = 2500 nM T37848 C6ZJ9E 44190581 IC50 = 3100 nM T37848 CMV52H 44191040 IC50 > 5000 nM T37848 C6SG0O 44192200 IC50 = 10000 nM T37848 C5L6WO 44194849 IC50 = 67000 nM T37848 CZ29JY 44205724 IC50 > 30000 nM T37848 C84YBA 44205825 IC50 > 50000 nM T37848 C5RL9M 44215838 IC50 = 30000 nM T37848 C7VWX5 44220300 IC50 > 10000 nM T37848 C2O0NL 44230575 IC50 > 20000 nM T37848 CX4YL8 44232522 IC50 > 10000 nM T37848 CQ13MH 44234032 IC50 > 50000 nM T37848 C7UY5F 44235863 IC50 > 10000 nM T37848 CX2W8Y 44236320 IC50 > 10000 nM T37848 C8LN0U 44236321 IC50 = 10000 nM T37848 CK4S5Y 44236322 IC50 < 10000 nM T37848 C4W0SH 44247585 IC50 > 40000 nM T37848 C43UTJ 44247586 IC50 = 24000 nM T37848 C7MY2N 44247806 IC50 > 10000 nM T37848 CDOA12 44249906 IC50 > 41000 nM T37848 C85DHY 44250284 IC50 > 5000 nM T37848 C8P2LE 44250288 IC50 > 10000 nM T37848 CLY1A3 44251218 IC50 > 25000 nM T37848 CNO97U 44255810 IC50 > 20000 nM T37848 C4XW9G 44266800 IC50 = 22000 nM T37848 C7ZYM4 44299404 IC50 > 50000 nM T37848 C5FQH4 44317319 IC50 = 6100 nM T37848 C3RN4G 44317321 IC50 = 6100 nM T37848 CZ5A4P 44317414 IC50 < 50 nM T37848 C7S2ZI 44340870 IC50 = 470 nM T37848 CE13FX 44341241 IC50 > 100000 nM T37848 CX65PH 44341461 IC50 = 39000 nM T37848 C0KD4U 44346053 IC50 > 2000 nM T37848 CH0O5Q 44346322 IC50 > 2000 nM T37848 C0E5KX 44346577 IC50 = 1100 nM T37848 C9U6WK 44346578 IC50 = 10000 nM T37848 C5OQ2K 44366980 IC50 > 100000 nM T37848 CKF5G6 44367711 IC50 = 37000 nM T37848 CW48BI 44367781 IC50 = 7900 nM T37848 CQ05NO 44380394 IC50 = 5000 nM T37848 C8J6QW 44380537 IC50 = 1000 nM T37848 C4T3JB 44380538 IC50 = 1000 nM T37848 C16VXA 44380625 IC50 = 100 nM T37848 C7DA2K 44380681 IC50 > 10000 nM T37848 CU2EP8 44380796 IC50 = 1000 nM T37848 CM6V4C 44388606 IC50 = 262000 nM T37848 CKV1H9 44388612 IC50 = 109000 nM T37848 CGU79D 44388657 IC50 = 77500 nM T37848 CAWG69 44390123 IC50 = 397 nM T37848 CDZH20 44390134 IC50 = 200 nM T37848 CIOY83 44390142 IC50 = 357 nM T37848 CDQ90V 44390161 IC50 = 140 nM T37848 CS5NY3 44390206 IC50 = 481 nM T37848 CT5DF2 44390231 IC50 = 750 nM T37848 CH1QM4 44390265 IC50 = 2200 nM T37848 CN91AI 44399944 IC50 = 600 nM T37848 C50MUR 44400121 IC50 = 300 nM T37848 C5YS3K 44400230 IC50 = 440 nM T37848 CLIK31 44400235 IC50 = 100 nM T37848 COVG03 44400245 IC50 = 380 nM T37848 C68TAQ 44400261 IC50 = 180 nM T37848 C4NUA0 44402523 IC50 > 30000 nM T37848 CUGE51 44403300 IC50 = 13000 nM T37848 C8V7OA 44410763 IC50 = 448 nM T37848 C0SXD3 44410799 IC50 = 6300 nM T37848 C3PYC4 44410807 IC50 = 5300 nM T37848 CB6H1M 44410808 IC50 = 7500 nM T37848 CM4Z0T 44410814 IC50 = 800 nM T37848 CR4HX5 44410840 IC50 = 8200 nM T37848 C73OZJ 44410841 IC50 = 8000 nM T37848 C3NED2 44410860 IC50 > 20000 nM T37848 C1EA6U 44410861 IC50 = 1700 nM T37848 CU5E6C 44410862 IC50 = 580 nM T37848 CR5Y0N 44410871 IC50 = 400 nM T37848 C8IV5K 44410881 IC50 = 7000 nM T37848 CBS59K 44411032 IC50 = 2270 nM T37848 CRU1S5 44411036 IC50 = 2150 nM T37848 C9J8MS 44411109 IC50 = 1010 nM T37848 CFA64M 44411110 IC50 > 20000 nM T37848 CD53XR 44411116 IC50 = 2100 nM T37848 C7KZV2 44414322 IC50 = 254 nM T37848 CJM06T 44414347 IC50 > 10000 nM T37848 CF8Q6Y 44414836 IC50 = 10000 nM T37848 CQ2D0O 44418482 IC50 > 25000 nM T37848 CX09NV 44418490 IC50 > 25000 nM T37848 CY2F3Q 44420235 IC50 > 10000 nM T37848 CH1R7M 44420600 IC50 > 10000 nM T37848 CU52GB 44425701 IC50 = 12000 nM T37848 CX8TR0 44425719 IC50 = 7500 nM T37848 C89EXO 44425789 IC50 = 35 nM T37848 C2AE6C 44425801 IC50 > 10000 nM T37848 CH04WE 44425802 IC50 = 1100 nM T37848 C9D4LQ 44425803 IC50 = 300 nM T37848 C52ZIS 44425809 IC50 = 2000 nM T37848 CU7YW1 44425810 IC50 = 6200 nM T37848 C0WVT1 44425811 IC50 = 1700 nM T37848 CE3A2G 44425817 IC50 > 10000 nM T37848 C1IVD0 44425837 IC50 > 10000 nM T37848 CAWL05 44428924 IC50 = 3580 nM T37848 CTB82G 44431744 IC50 > 50000 nM T37848 CL6B7S 44431775 IC50 > 50000 nM T37848 C3B7EG 44433262 IC50 = 120 nM T37848 CPRL53 44433263 IC50 = 220 nM T37848 CKX7P2 44433264 IC50 = 49000 nM T37848 CQ91YU 44433265 IC50 = 640 nM T37848 CJZ3P7 44433266 IC50 = 2700 nM T37848 CRP35K 44433267 IC50 = 480 nM T37848 CF3J7G 44433268 IC50 = 35000 nM T37848 C3ZIE0 44433269 IC50 = 8900 nM T37848 CN51TW 44433270 IC50 = 6300 nM T37848 CQ4X7E 44433271 IC50 = 650 nM T37848 C4O5HS 44433272 IC50 = 4800 nM T37848 CEA96F 44433273 IC50 = 11000 nM T37848 CED62W 44433274 IC50 = 32000 nM T37848 CI29CM 44433275 IC50 = 37000 nM T37848 CEN1M3 44433276 IC50 = 3400 nM T37848 C9KT3N 44433277 IC50 = 15000 nM T37848 CS2YQ7 44433278 IC50 = 720 nM T37848 C27GZL 44433279 IC50 > 50000 nM T37848 CB29IZ 44433282 IC50 = 21000 nM T37848 COX3A0 44433283 IC50 = 25000 nM T37848 CAE5J2 44433284 IC50 = 3600 nM T37848 C9U4FM 44433285 IC50 = 2300 nM T37848 CB6P5W 44433286 IC50 = 6500 nM T37848 C3R0EA 44433287 IC50 = 3600 nM T37848 CZN71T 44433288 IC50 = 15000 nM T37848 CR54CU 44433289 IC50 = 5300 nM T37848 C1M0JP 44433290 IC50 = 2900 nM T37848 C9ZT8U 44433291 IC50 = 8600 nM T37848 CI62TG 44433292 IC50 = 28000 nM T37848 CZ3I4N 44433293 IC50 = 2900 nM T37848 CZU4D1 44433294 IC50 = 6700 nM T37848 CS5TK4 44433295 IC50 = 6400 nM T37848 CYH7M2 44433296 IC50 = 5400 nM T37848 C7E4KR 44433297 IC50 = 1300 nM T37848 CPX57U 44433298 IC50 = 3400 nM T37848 CI2PC5 44433299 IC50 = 6900 nM T37848 C89WJP 44433300 IC50 = 15000 nM T37848 C9LM7U 44433789 IC50 = 18000 nM T37848 CWDJ93 44433797 IC50 = 11000 nM T37848 CU67NA 44433798 IC50 = 49000 nM T37848 CNU4B6 44433799 IC50 = 11000 nM T37848 C5V7WE 44433800 IC50 = 23000 nM T37848 CBP25Q 44433802 IC50 = 28000 nM T37848 CB1SD9 44433803 IC50 = 100000 nM T37848 C4Q2MH 44435366 IC50 = 400 nM T37848 CX51JK 44435367 IC50 = 400 nM T37848 C1SCL8 44435394 IC50 = 400 nM T37848 C8BAW3 44439731 IC50 = 2000 nM T37848 CP2G6L 44440493 IC50 = 6900 nM T37848 CXSQ75 44440525 IC50 = 28000 nM T37848 C2VAG9 44440645 IC50 > 10000 nM T37848 C08ZST 44440659 IC50 > 10000 nM T37848 CR3PM7 44440662 IC50 > 10000 nM T37848 CCSI57 44440665 IC50 > 10000 nM T37848 CV6MS8 44441997 IC50 = 1200 nM T37848 CDA0K3 44441998 IC50 = 1300 nM T37848 C6VF9N 44441999 IC50 = 5000 nM T37848 C5KPT0 44442000 IC50 = 3400 nM T37848 CSXU96 44442006 IC50 = 24300 nM T37848 CF2NQ0 44442007 IC50 = 300 nM T37848 CX5V1C 44442008 IC50 = 300 nM T37848 C41NKY 44442009 IC50 = 30000 nM T37848 CH97AI 44442010 IC50 = 10100 nM T37848 C31THS 44442011 IC50 = 15600 nM T37848 CPFY31 44442012 IC50 = 30000 nM T37848 CWTI80 44442013 IC50 = 800 nM T37848 C4NST7 44442014 IC50 = 500 nM T37848 C3YR2W 44442017 IC50 = 11000 nM T37848 CT0C4I 44443093 IC50 > 20000 nM T37848 CF1V8O 44443098 IC50 = 12000 nM T37848 CHZ48Q 44443101 IC50 = 9000 nM T37848 CQ53TV 44443130 IC50 > 19000 nM T37848 CEZ6U8 44443131 IC50 > 16000 nM T37848 CN4XZ6 44443132 IC50 > 9000 nM T37848 CV5CK0 44443532 IC50 = 1000 nM T37848 CVRZ54 44444647 IC50 = 6000 nM T37848 CBZ9S3 44444649 IC50 > 10000 nM T37848 CO51RA 44445723 IC50 > 100000 nM T37848 C84SBR 44445724 IC50 > 100000 nM T37848 C1A2QH 44445725 IC50 > 100000 nM T37848 C8C3RN 44446982 IC50 = 4700 nM T37848 CXB95D 44446986 IC50 = 4200 nM T37848 COD25M 44446990 IC50 = 300 nM T37848 CL92EJ 44446991 IC50 = 4700 nM T37848 C3QA8R 44446995 IC50 = 1800 nM T37848 C24BTK 44446997 IC50 < 30 nM T37848 C94ABT 44446998 IC50 > 30000 nM T37848 CBP6U4 44447000 IC50 = 16900 nM T37848 CK29XH 44447004 IC50 = 4000 nM T37848 CIR43Q 44447017 IC50 = 2600 nM T37848 C6AG0K 44447021 IC50 = 3100 nM T37848 CF7S4D 44447022 IC50 = 1200 nM T37848 CNYP84 44447024 IC50 = 300 nM T37848 C5NWH2 44447027 IC50 = 700 nM T37848 C82PEY 44447030 IC50 = 300 nM T37848 CD6FA4 44447033 IC50 = 300 nM T37848 C4BGZ1 44447036 IC50 = 600 nM T37848 CYH4O2 44447257 IC50 = 860 nM T37848 CHMJ82 44447262 IC50 = 980 nM T37848 C3B1OF 44447264 IC50 = 2430 nM T37848 C5C3YI 44447269 IC50 = 820 nM T37848 C5MT0J 44447277 IC50 = 1900 nM T37848 C7PB9V 44447278 IC50 = 1800 nM T37848 CQ7AT9 44447279 IC50 = 6000 nM T37848 CIY3T7 44447280 IC50 > 10000 nM T37848 CP7D3U 44447281 IC50 > 10000 nM T37848 CC71MI 44447282 IC50 = 1300 nM T37848 CEF81H 44447283 IC50 = 2400 nM T37848 CULB63 44447285 IC50 > 20000 nM T37848 CK4Q6O 44447286 IC50 = 4600 nM T37848 C0PT9W 44447287 IC50 = 6100 nM T37848 C5NKU9 44447288 IC50 = 3900 nM T37848 CY41VI 44447289 IC50 = 5300 nM T37848 CX8GC7 44447290 IC50 = 2000 nM T37848 CK6Q0S 44447291 IC50 = 810 nM T37848 CJM6O7 44447293 IC50 = 3400 nM T37848 CBC5F7 44447294 IC50 > 20000 nM T37848 CYB0L8 44447295 IC50 > 20000 nM T37848 CHS74Q 44447296 IC50 = 980 nM T37848 C5K8ZM 44447866 IC50 = 6100 nM T37848 C8W5YG 44447872 IC50 > 10000 nM T37848 CAOB06 44448056 IC50 = 1100 nM T37848 CY8RO4 44448772 IC50 = 770 nM T37848 C9K8EN 44448775 IC50 = 1400 nM T37848 CW7BG9 44448874 IC50 = 680 nM T37848 CR6TO5 44448876 IC50 = 1000 nM T37848 CF40AD 44448913 IC50 = 1300 nM T37848 C5OR0Q 44448947 IC50 = 2100 nM T37848 C15VTJ 44448976 IC50 = 2700 nM T37848 C1F2MP 44449004 IC50 = 6800 nM T37848 CL9M2D 44449052 IC50 = 1000 nM T37848 CL4H8Y 44449053 IC50 = 1200 nM T37848 C3L4XD 44449079 IC50 = 3900 nM T37848 C4T1MQ 44449106 IC50 = 1800 nM T37848 C9XZY1 44449107 IC50 = 730 nM T37848 CV31WQ 44449136 IC50 = 480 nM T37848 CA4DS0 44449171 IC50 = 1200 nM T37848 CA61WE 44449202 IC50 = 490 nM T37848 CC19LO 44449228 IC50 = 1100 nM T37848 C3RMF8 44449236 IC50 > 10000 nM T37848 C61KOC 44449479 IC50 = 6400 nM T37848 CUB12D 44449577 IC50 > 40000 nM T37848 CTLO32 44451459 IC50 = 12000 nM T37848 CW62HN 44451470 IC50 = 7500 nM T37848 C7WM5I 44451471 IC50 = 7800 nM T37848 CXRG25 44451484 IC50 = 17000 nM T37848 C4U8SK 44451494 IC50 > 20000 nM T37848 CZB82I 44451497 IC50 = 19000 nM T37848 CXPD58 44453913 IC50 > 40000 nM T37848 C9YUM3 44453941 IC50 = 20000 nM T37848 CPM4W2 44454303 IC50 = 5500 nM T37848 CD3HE5 44454670 IC50 > 10000 nM T37848 CJ6N1L 44454671 IC50 = 7000 nM T37848 C0MF7P 44454684 IC50 = 200 nM T37848 C9M3PR 44454697 IC50 = 1300 nM T37848 CL6KS1 44454834 IC50 > 5000 nM T37848 CC56ZN 44454845 IC50 = 800 nM T37848 CHY9A8 44454940 IC50 = 1800 nM T37848 CZ39GO 44455035 IC50 > 10000 nM T37848 CA8GN6 44456034 IC50 > 100000 nM T37848 CNGI92 44456070 IC50 > 100000 nM T37848 CU1R3D 44456109 IC50 > 100000 nM T37848 CQ27WK 44456229 IC50 > 100000 nM T37848 CPR06N 44456424 IC50 = 1000 nM T37848 CH82JM 44456599 IC50 = 1500 nM T37848 CWL42H 44457199 IC50 = 95 nM T37848 CGT38B 44462719 IC50 = 16000 nM T37848 CYQX20 44465025 IC50 = 620 nM T37848 C7UDS1 44467360 IC50 > 30000 nM T37848 C8C1VG 44467504 IC50 > 20000 nM T37848 C0CNQ3 44467506 IC50 > 20000 nM T37848 CL5XQ6 44467507 IC50 > 30000 nM T37848 C41RNH 44467574 IC50 > 30000 nM T37848 C8TIU2 44467575 IC50 > 30000 nM T37848 CM41YP 44467576 IC50 = 34100 nM T37848 CLU19G 44467711 IC50 = 30000 nM T37848 CVC68I 44467853 IC50 > 20000 nM T37848 C1ZBJ3 44469819 IC50 > 6000 nM T37848 C2QK4J 44472590 IC50 > 100000 nM T37848 CQ8C3F 44472591 IC50 = 96000 nM T37848 CWN95E 44472610 IC50 > 100000 nM T37848 C1H2ZT 44472612 IC50 > 100000 nM T37848 CC75ON 44473086 IC50 = 300 nM T37848 CUZ97H 44473093 IC50 = 900 nM T37848 CSFM32 44473094 IC50 = 400 nM T37848 C2OT5K 44473095 IC50 = 7000 nM T37848 C4H0DY 44473096 IC50 = 8000 nM T37848 C7S8OZ 44473097 IC50 = 87000 nM T37848 CO19AD 44473098 IC50 = 18000 nM T37848 CTP32R 44473099 IC50 = 18000 nM T37848 CJM1U2 44473400 IC50 = 1500 nM T37848 C3GYC0 44475943 IC50 >= 100000 nM T37848 CX9TJ4 44476890 IC50 = 48000 nM T37848 CNG6R4 44476952 IC50 = 1400 nM T37848 CY4MJ6 44478726 IC50 = 18000 nM T37848 C12HYU 44478952 IC50 = 130 nM T37848 CTK38R 44478953 IC50 = 270 nM T37848 CUA9F0 44512094 IC50 > 50000 nM T37848 C4M9FH 44512619 IC50 > 40000 nM T37848 CU80BP 44517743 IC50 > 30000 nM T37848 CS9H0L 44517795 IC50 > 50000 nM T37848 CKI82C 44518336 IC50 > 1000 nM T37848 CSO35V 44520546 IC50 = 501.19 nM T37848 CJCB39 44520861 IC50 = 7900 nM T37848 CJA36X 44533150 IC50 > 50000 nM T37848 CVZW52 44537923 IC50 > 50000 nM T37848 C9N1BU 44539192 IC50 > 20000 nM T37848 C14SNF 44539764 IC50 > 30000 nM T37848 CLMY52 44539967 IC50 > 10000 nM T37848 CMW56J 44539973 IC50 > 30000 nM T37848 C0RA9E 44540072 IC50 > 30000 nM T37848 CR19IH 44543858 IC50 = 15000 nM T37848 C05HEP 44543860 IC50 = 6000 nM T37848 C45ZHO 44543969 IC50 = 3000 nM T37848 C27TZY 44543970 IC50 = 8000 nM T37848 C25OXZ 44544094 IC50 = 4000 nM T37848 C7JIF6 44544321 IC50 = 15000 nM T37848 CK1Z8P 44545482 IC50 = 34000 nM T37848 CECD12 44547033 IC50 = 330 nM T37848 CX13MK 44547414 IC50 > 50000 nM T37848 CP6R2X 44551848 IC50 = 6000 nM T37848 C4RB7W 44555352 IC50 > 10000 nM T37848 C5EX1K 44555473 IC50 < 10000 nM T37848 CVJ8S4 44559524 IC50 = 98300 nM T37848 CCGE36 44559528 IC50 = 36400 nM T37848 C32AGV 44561123 IC50 = 3300 nM T37848 CG1W8A 44561157 IC50 = 4900 nM T37848 CXH86I 44561195 IC50 = 2100 nM T37848 CD7A4H 44561196 IC50 = 4600 nM T37848 C8HCR6 44561197 IC50 = 9100 nM T37848 C9HG8L 44561236 IC50 = 4200 nM T37848 CR5T0L 44561237 IC50 = 9000 nM T37848 CF21JK 44561238 IC50 = 2600 nM T37848 CMJ60R 44561239 IC50 = 2200 nM T37848 C0W4HQ 44561240 IC50 = 6400 nM T37848 C6A0TH 44561276 IC50 = 1000 nM T37848 CPW0S4 44561816 IC50 > 100000 nM T37848 CS7O8X 44564029 Ki < 50000000 nM T37848 CQ8UN1 44564037 Ki < 50000000 nM T37848 CU9J5W 44564565 IC50 > 100000 nM T37848 CV1IL5 44565796 IC50 > 10000 nM T37848 C8DUG3 44566070 EC50 = 3400 nM T37848 CJB91U 44568803 IC50 = 1800 nM T37848 CR7C6A 44568804 IC50 = 5600 nM T37848 C97CEZ 44568805 IC50 = 4000 nM T37848 CQ7SL3 44568819 IC50 = 4200 nM T37848 C1OVN0 44568820 IC50 = 5600 nM T37848 C4MNS3 44568821 IC50 = 10000 nM T37848 COPU28 44568925 IC50 > 25000 nM T37848 CSQ1F7 44568926 IC50 = 12000 nM T37848 C6QG1U 44568927 IC50 > 25000 nM T37848 CT2CX7 44568928 IC50 > 25000 nM T37848 CCV6K0 44568929 IC50 = 6000 nM T37848 C25LHW 44568941 IC50 > 25000 nM T37848 CK67DM 44568942 IC50 > 25000 nM T37848 C3PTD5 44568943 IC50 = 4500 nM T37848 C4CX6W 44568944 IC50 > 25000 nM T37848 CB5S9R 44569927 IC50 = 58000 nM T37848 C6Q5DK 44569945 IC50 = 700 nM T37848 CWLT20 44570180 IC50 = 320 nM T37848 CBET53 44570224 IC50 = 100000 nM T37848 CP32DL 44570256 IC50 > 100000 nM T37848 CVO8L1 44570275 IC50 = 500 nM T37848 C78BLW 44570364 IC50 = 7000 nM T37848 CQJ68M 44570365 IC50 = 6000 nM T37848 CR9YO2 44570410 IC50 = 1500 nM T37848 CJX16E 44570412 IC50 = 3000 nM T37848 CX8HP4 44570452 IC50 = 40000 nM T37848 CKON49 44570453 IC50 = 900 nM T37848 CPX08J 44570489 IC50 = 500 nM T37848 CE2BR6 44570490 IC50 = 8400 nM T37848 CF13PE 44570491 IC50 = 12000 nM T37848 C84ZAY 44570492 IC50 = 3500 nM T37848 CGB85R 44570528 IC50 = 4800 nM T37848 CH21FR 44573547 IC50 = 4900 nM T37848 CZ56HX 44574108 IC50 > 5000 nM T37848 CTA0G9 44576642 IC50 = 800 nM T37848 CLE52Y 44576643 IC50 = 9100 nM T37848 CV4HU0 44576644 IC50 = 48 nM T37848 C74QBS 44576645 IC50 = 120 nM T37848 CVZ2A9 44576655 IC50 = 670 nM T37848 C32ANR 44576656 IC50 = 20000 nM T37848 C38AKC 44576657 IC50 = 16000 nM T37848 C9IB4V 44576677 IC50 = 31000 nM T37848 CY1KQ8 44576678 IC50 = 130 nM T37848 CRS2A0 44576679 IC50 = 33000 nM T37848 CMZ6C1 44576680 IC50 > 50000 nM T37848 CSIH37 44576681 IC50 = 20000 nM T37848 CBKL21 44577683 IC50 = 12000 nM T37848 C01CYU 44578045 IC50 = 180 nM T37848 CFJB16 44578266 IC50 > 3000 nM T37848 CG80OC 44578914 IC50 > 50000 nM T37848 C7LAT0 44578954 IC50 > 50000 nM T37848 CBG04P 44578955 IC50 > 50000 nM T37848 CA3FO8 44578956 IC50 > 50000 nM T37848 CA16QJ 44578957 IC50 > 50000 nM T37848 CFH01N 44578958 IC50 > 50000 nM T37848 CMA26F 44578959 IC50 > 50000 nM T37848 C79PYS 44578960 IC50 > 50000 nM T37848 CF39ON 44578961 IC50 > 50000 nM T37848 CB2K9P 44578988 IC50 > 10000 nM T37848 C68JSG 44579085 IC50 = 12000 nM T37848 CVU2Z0 44579129 IC50 = 2500 nM T37848 CEH1N0 44579131 IC50 = 27000 nM T37848 CW69AF 44579132 IC50 = 39000 nM T37848 CM1PH0 44579133 IC50 = 22000 nM T37848 CL3J1S 44579180 IC50 = 12000 nM T37848 C4N2PZ 44579181 IC50 = 15000 nM T37848 C74XJR 44579182 IC50 = 7800 nM T37848 C4KI0B 44579189 IC50 > 50000 nM T37848 C1I0QG 44579190 IC50 > 50000 nM T37848 C6VFZ3 44579191 IC50 > 50000 nM T37848 C1O5ET 44579232 IC50 > 50000 nM T37848 CY8NJ4 44579233 IC50 > 50000 nM T37848 CSLC36 44579234 IC50 > 50000 nM T37848 CBK23W 44579235 IC50 > 50000 nM T37848 CS2KV6 44579236 IC50 > 50000 nM T37848 C60CAD 44579237 IC50 > 50000 nM T37848 CX85MD 44579273 IC50 > 50000 nM T37848 C0IP7C 44583234 IC50 > 10000 nM T37848 C6HTC1 44583235 IC50 > 10000 nM T37848 CZJU04 44583236 IC50 > 10000 nM T37848 C3TYW0 44583237 IC50 < 10000 nM T37848 CCL9R0 44583238 IC50 > 10000 nM T37848 COX7F1 44583287 IC50 < 10000 nM T37848 C5SI9Q 44583288 IC50 > 10000 nM T37848 CFT74N 44583289 IC50 > 10000 nM T37848 CC19TZ 44583290 IC50 > 10000 nM T37848 C90RAV 44583349 IC50 > 10000 nM T37848 CK81NJ 44583350 IC50 > 10000 nM T37848 C20VTN 44583351 IC50 > 10000 nM T37848 CD5U3A 44583352 IC50 > 10000 nM T37848 C9G7VT 44583353 IC50 > 10000 nM T37848 C6QF4O 44583354 IC50 > 10000 nM T37848 C48AQR 44583355 IC50 > 10000 nM T37848 CG5X0M 44583356 IC50 > 10000 nM T37848 CUG9Y0 44583357 IC50 > 10000 nM T37848 CRE9Q2 44583561 IC50 = 22000 nM T37848 C9AP1O 44583590 IC50 = 6500 nM T37848 CO6XB8 44583591 IC50 = 16000 nM T37848 CM6Y4F 44583614 IC50 = 4800 nM T37848 CR13XJ 44583631 IC50 = 3800 nM T37848 C53KBN 44583632 IC50 = 2900 nM T37848 CK27DJ 44583633 IC50 = 4200 nM T37848 C9EX2M 44583647 IC50 = 13000 nM T37848 C7K6YM 44583648 IC50 = 18000 nM T37848 CZ2D3P 44583663 IC50 = 62000 nM T37848 C5XD4S 44583664 IC50 = 3100 nM T37848 CKW9Y5 44583665 IC50 = 7700 nM T37848 CDZN40 44583666 IC50 = 700 nM T37848 C0IFL7 44583667 IC50 = 9200 nM T37848 CHR03D 44583679 IC50 = 31000 nM T37848 CZR8A3 44586731 IC50 = 800 nM T37848 CY2WG3 44587391 IC50 = 36000 nM T37848 CZ35WG 44587392 IC50 = 25000 nM T37848 CDIQ98 44587393 IC50 = 22000 nM T37848 C81XUZ 44587394 IC50 = 10000 nM T37848 C72XPL 44587398 IC50 = 42000 nM T37848 CAO71W 44587401 IC50 = 33000 nM T37848 CA7FG6 44587403 IC50 = 10000 nM T37848 C37JHB 44587404 IC50 = 22000 nM T37848 CSZ7D4 44587405 IC50 = 10000 nM T37848 C9RA0C 44589548 EC50 > 50000 nM T37848 CH54CO 44589824 IC50 = 720 nM T37848 C89LHN 44589825 IC50 = 3110 nM T37848 C94HFG 44590271 IC50 = 550 nM T37848 CH3CY9 44590272 IC50 = 870 nM T37848 CUB2R6 44590570 IC50 = 1300 nM T37848 CH97WM 44590571 IC50 = 1350 nM T37848 C70MSI 44593549 IC50 = 3000 nM T37848 CEFN61 44593613 IC50 = 350 nM T37848 CQ3U9E 44593614 IC50 = 36000 nM T37848 CIMG71 44593615 IC50 = 510 nM T37848 CCA7K5 44593648 IC50 > 50000 nM T37848 C64ZKC 44593664 IC50 > 10000 nM T37848 C01BFQ 44593665 IC50 > 10000 nM T37848 CE97GB 44596160 IC50 > 20000 nM T37848 COMB36 44601452 IC50 = 1100 nM T37848 C4ID9A 44602971 IC50 = 18000 nM T37848 C7I4EY 44603096 IC50 > 30000 nM T37848 C4MOE2 44603271 IC50 = 9000 nM T37848 C89VRG 44605616 IC50 = 1258.93 nM T37848 CZD25I 44605617 IC50 = 1258.93 nM T37848 CXQ19C 44610104 IC50 = 16000 nM T37848 C0WVZ1 44622338 IC50 > 30000 nM T37848 CL26YD 44622339 IC50 > 30000 nM T37848 CA7EQ2 44622340 IC50 > 30000 nM T37848 C23ORN 44622341 IC50 > 30000 nM T37848 C2JIX6 44622342 IC50 > 30000 nM T37848 CNI29G 44622416 IC50 > 30000 nM T37848 C9KUD5 44622417 IC50 > 30000 nM T37848 C4Q7JB 44622418 IC50 > 30000 nM T37848 C12SGH 44622499 IC50 > 30000 nM T37848 C2OUJ0 44624151 IC50 = 340 nM T37848 CT65UM 44624240 IC50 = 700 nM T37848 C7YOT9 44624488 IC50 > 50000 nM T37848 C0N6DO 44625908 IC50 = 11600 nM T37848 CXD90A 44625911 IC50 = 24100 nM T37848 C85ZIF 44626928 IC50 > 10000 nM T37848 C4BYG5 44626929 IC50 > 10000 nM T37848 CQE59L 44627133 IC50 > 10000 nM T37848 CDQ47G 44629236 IC50 > 25000 nM T37848 CH3SF9 44631836 IC50 > 27000 nM T37848 C1SYK4 44633765 Ki = 9500 nM T37848 CPG61Y 44718445 IC50 > 20000 nM T37848 C37AQP 44815590 IC50 > 10000 nM T37848 C3Q7BW 44816514 IC50 > 30000 nM T37848 C85DWU 44816692 IC50 = 18000 nM T37848 CJ0F5Q 44819015 IC50 = 4000 nM T37848 CN21OS 44819193 IC50 > 30000 nM T37848 CSEP-69 45102708 IC50 > 8000 nM T37848 C32YHG 45102733 IC50 = 29000 nM T37848 CGCZ64 45102767 IC50 > 50000 nM T37848 C7NFZ1 45110765 IC50 > 30000 nM T37848 CR6UW4 45112038 IC50 > 50000 nM T37848 CUL67Y 45202552 IC50 = 28200 nM T37848 C4IY8M 45256689 IC50 > 50000 nM T37848 C1K0ZH 45259193 IC50 = 10000 nM T37848 CB9QZ6 45263405 IC50 > 30000 nM T37848 CQ85WF 45263621 IC50 > 10000 nM T37848 CMJ1U7 45266443 IC50 > 80000 nM T37848 CUT2B4 45267348 IC50 > 10000 nM T37848 CI7KZ2 45267735 IC50 = 3220 nM T37848 CC5OP0 45267739 IC50 = 13400 nM T37848 C53DIE 45267853 IC50 < 15000 nM T37848 CJH3A2 45268206 IC50 > 10000 nM T37848 CULJ91 45268456 IC50 = 11000 nM T37848 C9B5EH 45268653 IC50 > 5000 nM T37848 C4WR0V 45269087 IC50 > 10000 nM T37848 CRPS25 45269096 IC50 > 10000 nM T37848 C7BNY6 45269104 IC50 > 10000 nM T37848 CB5O6V 45269307 IC50 > 30000 nM T37848 CS1Q2X 45269947 IC50 > 10000 nM T37848 C1BE5U 45269948 IC50 > 10000 nM T37848 CG1H9N 45269950 IC50 > 10000 nM T37848 C03ETI 45270148 IC50 > 30000 nM T37848 C4SXQ3 45270319 IC50 = 16500 nM T37848 C8GQ7J 45270330 IC50 > 5000 nM T37848 C48BMQ 45270339 IC50 > 5000 nM T37848 C1NT2M 45270771 IC50 > 10000 nM T37848 CA05IG 45270778 IC50 > 10000 nM T37848 CZ7MK9 45270788 IC50 > 10000 nM T37848 CY70SI 45270983 IC50 > 30000 nM T37848 C2XH3A 45270987 IC50 > 30000 nM T37848 CY70FL 45271134 IC50 = 2490 nM T37848 C18WQE 45271166 IC50 > 5000 nM T37848 C9TM2P 45271593 IC50 > 10000 nM T37848 C06YAD 45271599 IC50 > 10000 nM T37848 CG0I8P 45271610 IC50 > 10000 nM T37848 C6FBH0 45271618 IC50 < 10000 nM T37848 C2MKZ1 45272040 IC50 = 320 nM T37848 CU9C4I 45272046 IC50 > 5000 nM T37848 CAY8I7 45272070 IC50 > 5000 nM T37848 CB25TO 45272156 IC50 = 300 nM T37848 C71VIG 45272510 IC50 < 10000 nM T37848 C05EDY 45272511 IC50 > 10000 nM T37848 C35DUQ 45272700 IC50 > 30000 nM T37848 CKUI32 45272704 IC50 > 30000 nM T37848 C3GUS5 45272853 IC50 = 570 nM T37848 C62IGT 45272875 IC50 > 5000 nM T37848 C3GUK4 45272876 IC50 > 5000 nM T37848 CBE0M8 45272877 IC50 > 5000 nM T37848 CR04WH 45272878 IC50 > 5000 nM T37848 CZ7N8Q 45272889 IC50 > 5000 nM T37848 CK2B5U 45272890 IC50 > 5000 nM T37848 C8TC4R 45272894 IC50 = 72000 nM T37848 CA0SD1 45272895 IC50 > 5000 nM T37848 CD62AH 45273373 IC50 > 10000 nM T37848 CMN39U 45273380 IC50 > 10000 nM T37848 C3U7KT 45273637 IC50 > 30000 nM T37848 C3TZ8X 45273801 IC50 = 4400 nM T37848 CX9T5I 45273802 IC50 = 790 nM T37848 C5E2XR 45273828 IC50 > 5000 nM T37848 CZ71RN 45278805 IC50 > 20000 nM T37848 CYOW10 45377016 IC50 > 20000 nM T37848 C7D3LB 45377018 IC50 > 20000 nM T37848 C25PTU 45377580 IC50 > 20000 nM T37848 C8ELI4 45378010 IC50 > 20000 nM T37848 CMU6Z8 45379828 IC50 > 6000 nM T37848 CNQT48 45379947 IC50 > 10000 nM T37848 CLK8O9 45380748 IC50 > 20000 nM T37848 C84ORB 45380848 IC50 = 18000 nM T37848 C0CHF4 45482789 IC50 > 10000 nM T37848 CQB4T6 45483078 Ki = 30 nM T37848 C1FSA3 45483090 Ki = 1548.82 nM T37848 CXJ0R7 45483091 Ki = 316.23 nM T37848 C9E0ZU 45483092 Ki = 575.44 nM T37848 CR48CA 45483093 Ki = 70 nM T37848 CKQD19 45483106 Ki = 1010 nM T37848 CY91DC 45483132 Ki = 165.96 nM T37848 CZUI01 45484860 IC50 = 3200 nM T37848 C65ONH 45484861 IC50 = 1000 nM T37848 C6KC8V 45484873 IC50 > 5000 nM T37848 CVR40A 45484874 IC50 = 4200 nM T37848 CV78NM 45484881 IC50 > 5000 nM T37848 C5DEA7 45484892 IC50 = 2900 nM T37848 CXYK82 45484893 IC50 = 1200 nM T37848 CR8VF3 45484894 IC50 = 2600 nM T37848 C7TQ3Z 45484899 IC50 = 4900 nM T37848 CD7N4J 45484900 IC50 > 5000 nM T37848 CQ84RV 45484907 IC50 > 5000 nM T37848 C1K0IO 45484913 IC50 > 5000 nM T37848 C2J4VM 45484915 IC50 = 1900 nM T37848 CE6J7S 45484916 IC50 = 4800 nM T37848 CI4SP9 45484917 IC50 > 5000 nM T37848 CYA6U2 45484918 IC50 > 5000 nM T37848 CYWT18 45484919 IC50 > 5000 nM T37848 C1FZ3N 45484922 IC50 > 5000 nM T37848 CXD74W 45484923 IC50 > 5000 nM T37848 CDP3X6 45484930 IC50 > 5000 nM T37848 CQ90DC 45484931 IC50 > 5000 nM T37848 CQ3I9D 45484949 IC50 = 3700 nM T37848 CZU29D 45484950 IC50 = 4400 nM T37848 CW6M7Q 45484961 IC50 > 5000 nM T37848 C4TI0X 45484966 IC50 = 1700 nM T37848 CWNH93 45484967 IC50 = 1900 nM T37848 C5R0YZ 45484968 IC50 = 1600 nM T37848 C9E4UO 45484969 IC50 > 5000 nM T37848 CL2M1O 45486624 IC50 = 2030 nM T37848 CDME83 45487345 IC50 > 35000 nM T37848 CC94VU 45487544 IC50 = 2030 nM T37848 C8HR9I 45487545 IC50 = 890 nM T37848 CP68GR 45487546 IC50 = 820 nM T37848 C2M5ZP 45487547 IC50 = 3790 nM T37848 C0P8RJ 45487551 IC50 > 5000 nM T37848 C3D6FX 45487553 IC50 = 2840 nM T37848 C8KZS7 45487862 IC50 = 9100 nM T37848 C98RSQ 45487864 IC50 = 16000 nM T37848 CR0X4I 45487870 IC50 = 26000 nM T37848 CL32NJ 45488686 IC50 > 10000 nM T37848 C1UK8O 46174269 IC50 = 1400 nM T37848 C7UAT9 46174270 IC50 = 4700 nM T37848 C8EX7B 46175090 IC50 = 800 nM T37848 COJ4E0 46175091 IC50 = 600 nM T37848 C7CK6V 46178246 IC50 = 11400 nM T37848 CB4O9P 46190694 Ki = 5600 nM T37848 CPU02J 46190696 IC50 = 12605 nM T37848 CQ5SD4 46190876 IC50 = 400 nM T37848 CE74UZ 46191161 IC50 = 4600 nM T37848 CQDI48 46191427 IC50 > 20000 nM T37848 CAT9Z8 46191428 IC50 > 20000 nM T37848 CP08ZD 46191499 IC50 > 20000 nM T37848 C0ET7O 46191501 IC50 > 20000 nM T37848 C4HSX5 46191502 IC50 > 20000 nM T37848 CSD13A 46191565 IC50 > 20000 nM T37848 CXIC58 46191567 IC50 = 20000 nM T37848 C71CGU 46191622 IC50 = 1000 nM T37848 CFYP54 46203897 IC50 = 3000 nM T37848 C21ICG 46212134 IC50 = 25400 nM T37848 CN3BE0 46212588 IC50 = 5000 nM T37848 CC9X1M 46213938 IC50 = 21800 nM T37848 CPF0J9 46214673 IC50 > 30000 nM T37848 CAX31B 46216689 IC50 > 15000 nM T37848 CL51NF 46216732 IC50 > 10000 nM T37848 CZJL95 46216733 IC50 > 10000 nM T37848 C5AY6M 46220498 IC50 > 10000 nM T37848 CSWY60 46225572 IC50 = 200 nM T37848 CS9GL5 46225573 IC50 = 100 nM T37848 CB5H9C 46225574 IC50 = 1300 nM T37848 C8M1DT 46225589 IC50 = 16 nM T37848 C60XUQ 46226079 IC50 = 100 nM T37848 C5PCH8 46226080 IC50 = 1000 nM T37848 C6UD1Y 46226095 IC50 = 790 nM T37848 C7IF4T 46226096 IC50 = 630 nM T37848 CUDZ46 46226135 IC50 = 5000 nM T37848 C0P4CT 46226136 IC50 = 500 nM T37848 CPH49S 46226137 IC50 = 1600 nM T37848 CM5X8B 46226156 IC50 = 4000 nM T37848 C64TVL 46226417 IC50 = 630 nM T37848 C1DO4U 46230960 IC50 = 8200 nM T37848 C59XOB 46230961 IC50 > 10000 nM T37848 C9EGU1 46230962 IC50 > 10000 nM T37848 C7G3TB 46231012 IC50 > 10000 nM T37848 C1J0WY 46231013 IC50 > 10000 nM T37848 CALC10 46231014 IC50 > 10000 nM T37848 C2FVA8 46231075 IC50 = 5000 nM T37848 CA3R5W 46231076 IC50 > 10000 nM T37848 CSZ2F6 46231077 IC50 > 10000 nM T37848 CVL6C0 46231146 IC50 = 7900 nM T37848 C8W4VL 46231147 IC50 = 8700 nM T37848 CRTO63 46231148 IC50 > 10000 nM T37848 CZ6C0S 46231149 IC50 > 10000 nM T37848 C80DAS 46231312 IC50 < 10000 nM T37848 CY5T7B 46232544 IC50 >= 16000 nM T37848 CTCG36 46232545 IC50 >= 8000 nM T37848 CVJU38 46233842 IC50 = 4200 nM T37848 CQ9A7L 46234188 IC50 > 30000 nM T37848 C94GCA 46234349 IC50 > 30000 nM T37848 C8PZU1 46235580 IC50 = 8.8 nM T37848 C7OB2G 46235733 IC50 = 9170 nM T37848 CIGB53 46237137 IC50 > 12 ug.mL-1 T37848 C0ZF4Y 46237255 IC50 = 2345 nM T37848 C8DYQ4 46237257 IC50 = 923 nM T37848 C0NEW2 46237259 IC50 = 1628 nM T37848 C9M6LO 46237408 IC50 = 275 nM T37848 CM82RF 46239494 IC50 = 7000 nM T37848 CQX93F 46398805 IC50 > 10000 nM T37848 CJ2D3O 46701015 IC50 > 5000 nM T37848 CM04ZI 46701016 IC50 = 12700 nM T37848 C0JWP5 46701017 IC50 > 25000 nM T37848 C5H0MJ 46701086 IC50 = 8390 nM T37848 C9HWI7 46701087 IC50 = 12800 nM T37848 CVE5O1 46701088 IC50 = 5280 nM T37848 C1VPM0 46701089 IC50 = 6500 nM T37848 CQ8B6R 46701090 IC50 > 5000 nM T37848 C6C0FS 46701091 IC50 > 5000 nM T37848 CMA4U3 46830115 Ki = 28.84 nM T37848 CC68WI 46830289 IC50 > 10000 nM T37848 C5TC2S 46830335 IC50 > 10000 nM T37848 C1K7FL 46830336 IC50 > 10000 nM T37848 CU5K1G 46834296 IC50 > 100000 nM T37848 C2M9XO 46835914 IC50 > 40000 nM T37848 C9CR0E 46835922 IC50 > 40000 nM T37848 C1L0GS 46840949 IC50 = 505 nM T37848 C4C0ED 46840950 IC50 = 827 nM T37848 CI1YK3 46841216 IC50 = 1271 nM T37848 CD8M3F 46841499 IC50 = 427 nM T37848 CO76ID 46841501 IC50 = 1058 nM T37848 CS5EJ1 46841648 IC50 = 12239 nM T37848 CRE97F 46841787 IC50 > 11248 nM T37848 COV0Q3 46841788 IC50 > 30000 nM T37848 C2OWF8 46841789 IC50 > 30000 nM T37848 C1N4KX 46842383 IC50 > 10000 nM T37848 CO1BZ7 46847258 IC50 = 10000 nM T37848 CPE23Q 46850145 IC50 > 20000 nM T37848 C2UYK7 46850264 IC50 > 50000 nM T37848 CD04SA 46852212 IC50 > 3000 nM T37848 CT6MJ2 46852951 IC50 > 50000 nM T37848 CBZE98 46853681 IC50 > 30000 nM T37848 CM58VK 46853747 IC50 = 7900 nM T37848 CO8C4F 46853748 IC50 = 2000 nM T37848 CUV83E 46854605 IC50 = 730 nM T37848 CIA08B 46854608 IC50 = 464 nM T37848 CWJ3F1 46854758 IC50 = 1330 nM T37848 CKRQ67 46854759 IC50 = 1770 nM T37848 CO31WX 46861576 IC50 = 8700 nM T37848 CC36NU 46861797 IC50 > 30000 nM T37848 CL5F9S 46861803 IC50 = 15000 nM T37848 CP6DN0 46861858 IC50 > 5000 nM T37848 C5VOF1 46861859 IC50 > 5000 nM T37848 CW1FS9 46861860 IC50 > 5000 nM T37848 CYC06D 46862027 IC50 = 2700 nM T37848 C9WY1K 46862028 IC50 = 31000 nM T37848 CO58RU 46862029 IC50 = 14000 nM T37848 CTVI92 46862134 IC50 = 2900 nM T37848 C78XDY 46862135 IC50 = 200 nM T37848 C4EY9T 46864494 IC50 > 40000 nM T37848 C0EG8P 46865563 IC50 = 10000 nM T37848 CC5KR7 46865978 IC50 > 10000 nM T37848 C9T0ZE 46866390 IC50 = 3500 nM T37848 CO3P0J 46866604 IC50 > 30000 nM T37848 CDG7J2 46868944 IC50 = 13500 nM T37848 CV0C3Y 46869239 IC50 = 6300 nM T37848 CO7N4V 46869440 IC50 > 20000 nM T37848 C56YTJ 46869566 IC50 = 12000 nM T37848 C0LRS2 46869760 IC50 = 2000 nM T37848 C8OY4U 46869951 IC50 > 30000 nM T37848 CLVI62 46879428 IC50 = 8800 nM T37848 CL2A4H 46879430 IC50 = 12000 nM T37848 C9VRO6 46879432 IC50 = 3100 nM T37848 CFH9W8 46879490 IC50 = 9600 nM T37848 CG68BI 46879549 IC50 = 90000 nM T37848 C9H1PK 46879550 IC50 = 7700 nM T37848 CB02YQ 46879551 IC50 = 1000 nM T37848 CCM7T2 46879552 IC50 = 22000 nM T37848 C7EHZ9 46879553 IC50 = 1300 nM T37848 CVI5O7 46879596 IC50 = 1600 nM T37848 CL05QN 46879597 IC50 = 2900 nM T37848 CYK18D 46879598 IC50 = 5600 nM T37848 CG9N6P 46879643 IC50 = 2400 nM T37848 CL8K6G 46880059 IC50 = 1900 nM T37848 CGH8L6 46880060 IC50 = 1300 nM T37848 CMA1P8 46880062 IC50 = 1000 nM T37848 CCK8A9 46880206 IC50 = 1600 nM T37848 C4BH9E 46882458 IC50 = 800 nM T37848 CQN87I 46882521 IC50 < 100 nM T37848 CRU1P2 46882874 IC50 > 10000 nM T37848 CYU8X6 46882875 IC50 < 10000 nM T37848 CX5CZ7 46882876 IC50 > 10000 nM T37848 C0FM2D 46882917 IC50 < 10000 nM T37848 CC1VO9 46882918 IC50 > 10000 nM T37848 C27RIV 46882919 IC50 > 10000 nM T37848 CE3O7D 46882949 IC50 > 10000 nM T37848 CHS1X0 46882950 IC50 < 10000 nM T37848 C3S9WE 46882951 IC50 > 10000 nM T37848 C3A1ZF 46882969 IC50 < 10000 nM T37848 CG3D0K 46882971 IC50 > 10000 nM T37848 CD7XA2 46882972 IC50 = 10000 nM T37848 CY5CW2 46882973 IC50 < 10000 nM T37848 C3ZPY7 46882986 IC50 > 10000 nM T37848 CKX8N2 46882987 IC50 > 10000 nM T37848 CG81CZ 46882988 IC50 > 10000 nM T37848 CP87CA 46883032 IC50 > 10000 nM T37848 CWU4T2 46883033 IC50 > 10000 nM T37848 C41RYD 46883034 IC50 > 10000 nM T37848 C3SQ2Z 46883035 IC50 > 10000 nM T37848 C0YZQ4 46883193 IC50 = 148 nM T37848 C7QX1S 46883194 IC50 = 90 nM T37848 C7DW3J 46883195 IC50 = 99 nM T37848 CSK3D5 46883196 IC50 = 65 nM T37848 CTVR02 46883197 IC50 = 110 nM T37848 C84SBC 46883198 IC50 = 100 nM T37848 C5EQB3 46883332 IC50 = 150 nM T37848 C6AI9B 46883333 IC50 = 110 nM T37848 CC50SV 46883334 IC50 = 110 nM T37848 CGZ52X 46883335 IC50 = 110 nM T37848 CGHM80 46883336 IC50 = 90 nM T37848 C2TC6H 46883337 IC50 = 67 nM T37848 CPR1N0 46883338 IC50 = 52 nM T37848 CWIN84 46883339 IC50 = 50 nM T37848 CJ90ET 46883340 IC50 = 135 nM T37848 C4ZX7N 46883341 IC50 = 87 nM T37848 CG7V1X 46883342 IC50 = 60 nM T37848 C1SC2E 46883343 IC50 = 50 nM T37848 CON39D 46883344 IC50 = 66 nM T37848 C0IW5K 46883345 IC50 = 49 nM T37848 C0S9ZY 46883346 IC50 = 66 nM T37848 CEG3S8 46883347 IC50 = 70 nM T37848 C7JWA9 46883369 IC50 > 3000 nM T37848 CO81JH 46883370 IC50 > 3000 nM T37848 CY35QT 46883371 IC50 = 1790 nM T37848 CI9FQ3 46883372 IC50 = 1330 nM T37848 CRLV61 46883373 IC50 = 136 nM T37848 C85MJW 46883397 IC50 = 88 nM T37848 C32RYS 46883398 IC50 = 66 nM T37848 C32AGP 46883399 IC50 = 135 nM T37848 CQL8U5 46883400 IC50 = 91 nM T37848 C5T2VX 46883401 IC50 = 300 nM T37848 C3W6BS 46883402 IC50 = 274 nM T37848 CVW81Y 46883435 IC50 = 348 nM T37848 CKJA72 46883436 IC50 = 741 nM T37848 C2R3CQ 46883437 IC50 = 3000 nM T37848 CH6WY4 46883438 IC50 > 300 nM T37848 CS51UC 46883473 IC50 < 10000 nM T37848 CL0S4B 46883474 IC50 > 10000 nM T37848 C0K5ZJ 46883508 IC50 < 10000 nM T37848 CMNJ24 46883509 IC50 < 10000 nM T37848 CF4VC1 46883510 IC50 < 10000 nM T37848 CN5C0Y 46883798 IC50 = 130 nM T37848 CTLN53 46883849 IC50 = 1300 nM T37848 CW6A9I 46884062 IC50 > 10000 nM T37848 C04JMO 46884063 IC50 > 10000 nM T37848 CR1Z8E 46884119 IC50 > 10000 nM T37848 CR0CQ9 46884120 IC50 > 10000 nM T37848 C9OYT5 46884152 IC50 > 10000 nM T37848 CCI32B 46884153 IC50 > 10000 nM T37848 C2JQE7 46884154 IC50 > 10000 nM T37848 C20HET 46884155 IC50 > 10000 nM T37848 C0HYN3 46884200 IC50 > 10000 nM T37848 CM6A8S 46884201 IC50 > 10000 nM T37848 CW94IK 46884202 IC50 > 10000 nM T37848 C3QT0U 46884239 IC50 = 5200 nM T37848 CB9O4H 46884365 Ki = 239.88 nM T37848 CKQZ62 46884411 Ki = 1778.28 nM T37848 C0ZL6F 46884412 Ki = 69.18 nM T37848 CU3BG6 46884668 IC50 > 10000 nM T37848 CPG14Q 46884669 IC50 > 10000 nM T37848 C7R9AK 46884670 IC50 > 10000 nM T37848 C64KNW 46884698 IC50 > 10000 nM T37848 C0ASK4 46884699 IC50 > 10000 nM T37848 CYNU85 46884731 IC50 > 10000 nM T37848 CJ6O8D 46884732 IC50 > 10000 nM T37848 C9QT7G 46884733 IC50 > 10000 nM T37848 CL6Z7Q 46884734 IC50 > 10000 nM T37848 C6PRX8 46884735 IC50 > 10000 nM T37848 CWK8I4 46884736 IC50 > 10000 nM T37848 C1A7XY 46884865 IC50 = 1200 nM T37848 CL0UV1 46884866 IC50 = 9100 nM T37848 CAG7P4 46884914 IC50 > 30000 nM T37848 C3MSG2 46885027 IC50 > 10000 nM T37848 CB7XI0 46885213 IC50 > 10000 nM T37848 CM76UZ 46888550 IC50 > 12 ug.mL-1 T37848 CZBL19 46888785 IC50 > 5000 nM T37848 CK3B2R 46888786 IC50 > 5000 nM T37848 C46QKX 46888787 IC50 > 5000 nM T37848 CJS87P 46888788 IC50 > 5000 nM T37848 C98ROS 46888789 IC50 > 5000 nM T37848 CNIH96 46888798 IC50 = 580 nM T37848 C08PXR 46888799 IC50 = 420 nM T37848 C9RXL8 46888825 IC50 > 5000 nM T37848 CHN7W1 46888826 IC50 > 5000 nM T37848 C46PXH 46888827 IC50 = 3300 nM T37848 CR42EN 46888828 IC50 > 5000 nM T37848 C5K7WG 46888836 IC50 = 2700 nM T37848 CY0ZJ7 46888837 IC50 = 650 nM T37848 C0D7BW 46888838 IC50 = 730 nM T37848 C3CT9F 46888839 IC50 = 270 nM T37848 C3B2QN 46888853 IC50 > 5000 nM T37848 C94FRI 46888854 IC50 > 5000 nM T37848 C30FVT 46888855 IC50 > 5000 nM T37848 C4Q2MA 46888856 IC50 > 5000 nM T37848 CJK1Z5 46888857 IC50 > 5000 nM T37848 CP73VU 46888864 IC50 = 300 nM T37848 CT7FM8 46888865 IC50 = 8400 nM T37848 CPJ73I 46888866 IC50 = 2900 nM T37848 CDBG34 46888867 IC50 = 2200 nM T37848 CL15PQ 46888898 IC50 = 5800 nM T37848 CPJN75 46888899 IC50 = 5200 nM T37848 CX92WH 46889257 IC50 > 5000 nM T37848 C01DMO 46889258 IC50 > 5000 nM T37848 CX18GT 46889932 IC50 > 10000 nM T37848 CQR58G 46892601 IC50 = 450 nM T37848 CIX16G 46892972 IC50 = 2200 nM T37848 CK6Z7P 46892975 IC50 = 1360 nM T37848 CS4XV6 46892977 IC50 = 760 nM T37848 C98JRZ 46893358 IC50 = 480 nM T37848 CZ90FC 46894119 IC50 = 5810 nM T37848 CC4GA0 46895367 IC50 = 3800 nM T37848 C90NYX 46896338 IC50 = 14000 nM T37848 CC9FZ0 46898063 IC50 > 20 nM T37848 C1JSH9 46899637 IC50 > 10000 nM T37848 CV3LP2 46899639 IC50 > 6000 nM T37848 CGHZ15 46899640 IC50 > 10000 nM T37848 CWR9M5 46900138 IC50 > 10000 nM T37848 CGN7Q8 46900139 IC50 > 10000 nM T37848 C40ZJO 46900451 IC50 < 4000 nM T37848 CNC02A 46900453 IC50 < 4000 nM T37848 CTCH14 46900455 IC50 < 4000 nM T37848 CP41AQ 46900457 IC50 = 100 nM T37848 CR3L4I 46900459 IC50 > 10000 nM T37848 CK17PA 46900606 IC50 > 5000 nM T37848 C1NAX4 46900612 IC50 > 5000 nM T37848 CXD9S3 46900776 IC50 > 10000 nM T37848 C8I7SJ 46900778 IC50 = 4000 nM T37848 C7QDM9 46900782 IC50 > 8000 nM T37848 C15FMY 46900954 IC50 > 7000 nM T37848 C7T2GX 46909057 IC50 > 50000 nM T37848 C3JCB1 46911060 IC50 > 50000 nM T37848 C4WXU5 46911119 IC50 = 1100 nM T37848 C2YM9P 46911173 IC50 = 1000 nM T37848 CHUV97 46911229 IC50 > 5000 nM T37848 C9SZ2X 46911333 IC50 < 68 nM T37848 CXJ7M5 46911719 IC50 = 8440 nM T37848 CA2GO4 46911720 IC50 = 9620 nM T37848 C1VA0B 46912953 IC50 > 5000 nM T37848 CN9L7G 46916268 IC50 > 10000 nM T37848 CR5OZ8 46916382 IC50 = 900 nM T37848 CLV1W2 46918487 IC50 = 5500 nM T37848 CJ3FM4 46925833 IC50 = 12860 nM T37848 C65QAB 46927297 IC50 > 10000 nM T37848 CM9UR2 46927440 IC50 = 800 nM T37848 C8GAI9 46927903 IC50 > 10000 nM T37848 C1TQV7 46927949 IC50 = 1900 nM T37848 C47HDL 46929447 IC50 = 17000 nM T37848 CSDO60 46929548 IC50 = 6500 nM T37848 C6F2MP 46929551 IC50 = 270 nM T37848 CZJ2G8 46929554 IC50 = 350 nM T37848 C3D7FL 46931619 IC50 = 20000 nM T37848 CKO76R 46931815 IC50 > 5000 nM T37848 C2M1KO 46932044 IC50 = 3000 nM T37848 C3QLC4 46932045 IC50 = 8000 nM T37848 CC91MK 46932046 IC50 = 7000 nM T37848 CQ91FA 46932047 IC50 = 15000 nM T37848 C70QIV 46932048 IC50 = 19000 nM T37848 CYCF24 46932049 IC50 = 18000 nM T37848 C3O4MA 46932136 IC50 = 20000 nM T37848 CF9YV2 46932138 IC50 > 50000 nM T37848 COL7J6 46932139 IC50 = 45000 nM T37848 CSMK50 46932141 IC50 = 32000 nM T37848 C29RXO 46932234 IC50 = 28000 nM T37848 CC0F4D 46932235 IC50 = 8000 nM T37848 C8QB4Z 46932237 IC50 = 17000 nM T37848 CJ0VB4 46932297 IC50 > 10000 nM T37848 CG2J9V 46932512 IC50 > 50000 nM T37848 C2VZ7Q 46932514 IC50 = 13000 nM T37848 C4PW3A 46932704 IC50 > 50000 nM T37848 CV98OS 46933385 IC50 > 30000 nM T37848 C0J8WS 46933530 IC50 = 30000 nM T37848 CJK53D 46933697 IC50 > 100000 nM T37848 CU90MG 46938037 IC50 > 20000000 nM T37848 CX2U5I 46938097 IC50 > 20000000 nM T37848 C47QBL 46938101 IC50 > 20000000 nM T37848 C9DLV2 46945057 IC50 > 50000 nM T37848 C03KOR 46945859 IC50 = 120 nM T37848 CZ0G6A 46947062 IC50 = 22680 nM T37848 CF14PE 46947264 IC50 > 30000 nM T37848 CX6NK2 47144386 IC50 = 400 nM T37848 CBV0H3 49765039 IC50 = 3500 nM T37848 CWU2R3 49773361 IC50 > 40000 nM T37848 C9RI3L 49780809 IC50 > 4000 nM T37848 CYL65E 49781476 IC50 > 10000 nM T37848 C2L7OT 49784695 IC50 = 40 nM T37848 CV4X7L 49787166 Ki = 990 nM T37848 CY1OJ5 49797177 IC50 > 30000 nM T37848 CQVG17 49798349 IC50 = 10000 nM T37848 C62VRQ 49798437 IC50 = 20417.38 nM T37848 CY90CD 49798461 IC50 = 19498.45 nM T37848 CF8J6E 49798462 IC50 = 436.52 nM T37848 CIC9S5 49799473 IC50 = 17650 nM T37848 C02EUQ 49800098 IC50 > 10000 nM T37848 C9YSF2 49800475 IC50 = 17000 nM T37848 CD8KX3 49804491 IC50 > 30000 nM T37848 CET89N 49822116 IC50 > 20000 nM T37848 CJ3SU6 49830359 IC50 = 2700 nM T37848 CVS85M 49831162 IC50 = 5000 nM T37848 CTP13K 49831178 IC50 = 4 nM T37848 C76XBM 49834039 IC50 = 3200 nM T37848 CGO57N 49834218 IC50 > 10000 nM T37848 COM5Q7 49836030 IC50 = 20200 nM T37848 CDO7I4 49836293 IC50 = 1100 nM T37848 CT7CV0 49836295 IC50 > 10000 nM T37848 CYJW87 49836299 IC50 > 10000 nM T37848 C8E6WA 49836410 IC50 > 10000 nM T37848 CNM9X8 49836528 IC50 > 10000 nM T37848 COK75S 49836633 IC50 > 10000 nM T37848 CB81YG 49836637 IC50 > 10000 nM T37848 CD8GN9 49837170 EC50 = 23000 nM T37848 CB71TA 49837867 IC50 > 50000 nM T37848 CZQC64 49837869 IC50 = 39000 nM T37848 CVNA15 49837870 IC50 = 37000 nM T37848 C9L3XR 49838879 IC50 > 13000 nM T37848 C06MKW 49839561 IC50 > 10000 nM T37848 C3DN7U 49843520 IC50 > 10000 nM T37848 CY46CB 49843532 IC50 > 50000 nM T37848 CU63QR 49847377 IC50 > 50000 nM T37848 CZT4I8 49847378 IC50 > 50000 nM T37848 CA72PE 49847379 IC50 > 50000 nM T37848 C8KQB9 49848139 IC50 > 10000 nM T37848 C4V7EW 49848258 IC50 > 10000 nM T37848 C4BXP1 49848557 IC50 > 50000 nM T37848 CQ32CR 49848656 IC50 > 10000 nM T37848 CP8TS6 49848895 IC50 > 50000 nM T37848 C9COF5 49848896 IC50 > 50000 nM T37848 CK0B1G 49848897 IC50 > 50000 nM T37848 CP61VJ 49849002 IC50 > 50000 nM T37848 CBM62Z 49849007 IC50 > 50000 nM T37848 C05SEW 49849008 IC50 > 50000 nM T37848 CF64IJ 49849120 IC50 > 50000 nM T37848 CC9EB4 49849122 IC50 > 50000 nM T37848 C2ORV5 49849123 IC50 > 50000 nM T37848 CTR7Q0 49850345 IC50 > 50118.72 nM T37848 C51QVH 49854023 IC50 = 40000 nM T37848 C8LBU5 49855513 IC50 > 30000 nM T37848 C5LY6T 49855593 IC50 = 10000 nM T37848 CQ0L4M 49856084 IC50 > 30000 nM T37848 C9TO2S 49856484 IC50 > 8900 nM T37848 C0N7RV 49856926 IC50 > 50000 nM T37848 C6POK9 49856931 IC50 > 50000 nM T37848 C9J7LZ 49857227 IC50 = 200 nM T37848 CC8VZ4 49857811 IC50 > 30000 nM T37848 CZO5D6 49857998 IC50 > 30000 nM T37848 CXT41G 49862010 IC50 = 6500 nM T37848 COS71Z 49862053 IC50 = 6800 nM T37848 CPL5O8 49862055 IC50 = 5900 nM T37848 C2H9XC 49862090 IC50 = 1100 nM T37848 C4RNH2 49862091 IC50 = 1900 nM T37848 CY9QB4 49862092 IC50 = 2800 nM T37848 CC6NY3 49862093 IC50 = 3500 nM T37848 C6MP7Y 49862094 IC50 = 3400 nM T37848 CK8M2Y 49862095 IC50 = 1000 nM T37848 CDK7E2 49862126 IC50 = 2100 nM T37848 CKO54S 49862127 IC50 = 1900 nM T37848 C3O5IR 49862128 IC50 = 900 nM T37848 C9PCE3 49862155 IC50 >= 7000 nM T37848 CM43HV 49862547 IC50 < 68 nM T37848 CFDH59 49862548 IC50 = 100 nM T37848 CNIA98 49862549 IC50 < 68 nM T37848 CKY2J9 49862550 IC50 < 68 nM T37848 CGU86D 49862599 IC50 < 68 nM T37848 CS4IP9 49862601 IC50 < 68 nM T37848 C63XUS 49862602 IC50 < 68 nM T37848 C6O7JQ 49862603 IC50 < 68 nM T37848 C8G7FR 49862604 IC50 < 68 nM T37848 CI41BU 49862643 IC50 < 100 nM T37848 C6O4ZK 49862647 IC50 = 4300 nM T37848 CP5D8Q 49862650 IC50 < 68 nM T37848 C6X0JA 49862651 IC50 < 68 nM T37848 C7BTK9 49862652 IC50 < 68 nM T37848 C79MQZ 49862653 IC50 = 900 nM T37848 CL8DR6 49862654 IC50 < 68 nM T37848 C10CAN 49862783 IC50 = 200 nM T37848 CGYM04 49864794 IC50 = 9500 nM T37848 C1I5PF 49864901 IC50 = 7500 nM T37848 CA4H2I 49864902 IC50 = 1500 nM T37848 CNFL69 49864903 IC50 > 30000 nM T37848 CY7U2X 49864936 IC50 = 11000 nM T37848 C8P2HI 49864937 IC50 = 13500 nM T37848 C8X3SL 49864938 IC50 = 6000 nM T37848 C2RN6C 49864988 IC50 = 9000 nM T37848 C59QLI 49864989 IC50 = 10600 nM T37848 CD29IW 49865043 IC50 > 30000 nM T37848 C6XT5M 49865104 IC50 = 400 nM T37848 CBMQ90 49865105 IC50 = 500 nM T37848 CMS6R4 49865106 IC50 = 300 nM T37848 C0Y5ZU 49865137 IC50 > 20 nM T37848 C6GJ0L 49865162 IC50 = 400 nM T37848 CA0RS7 49865163 IC50 = 200 nM T37848 C3WTC1 49865164 IC50 = 400 nM T37848 CG98LM 49865191 IC50 > 20 nM T37848 CR4F9G 49865290 IC50 > 50000 nM T37848 C0S8XD 49865953 IC50 = 51000 nM T37848 CMV6Y2 49868651 IC50 > 40000 nM T37848 C5OY7B 49872246 IC50 = 19000 nM T37848 C7GR0H 49872381 IC50 = 6940 nM T37848 CD1X3U 49872384 IC50 > 10000 nM T37848 C60RMP 49872483 IC50 = 25400 nM T37848 CV5BF3 49872645 IC50 = 14000 nM T37848 CN97FO 49872646 IC50 > 27000 nM T37848 CO0Y6K 49872677 IC50 > 10000 nM T37848 CD6P5R 49872735 IC50 > 27000 nM T37848 CL64NB 49872737 IC50 > 27000 nM T37848 CJWE29 49872771 IC50 > 10000 nM T37848 CK9VE4 49872772 IC50 > 10000 nM T37848 CFP14Q 49872867 IC50 > 10000 nM T37848 C83CTW 49872868 IC50 > 10000 nM T37848 CLB34U 49872872 IC50 > 10000 nM T37848 CAM1D0 49873181 IC50 > 10000 nM T37848 CV1L4P 49873242 IC50 > 27000 nM T37848 C5BA2V 49873243 IC50 > 27000 nM T37848 CSN45W 49873329 IC50 > 27000 nM T37848 CD2FS9 50898445 IC50 = 11.3 nM T37848 C8LA9S 50899467 IC50 > 30 nM T37848 CU7TK4 50899749 IC50 > 20000 nM T37848 CZ9UD6 50901657 IC50 = 2 nM T37848 C1R5UC 50905013 IC50 = 5000 nM T37848 C1N4YP 50908737 IC50 = 12000 nM T37848 CENW12 50925404 IC50 > 100000 nM T37848 CK1CD3 50925423 IC50 = 11900 nM T37848 CMF7T6 50925457 IC50 > 5000 nM T37848 C2GTE4 50938548 IC50 = 4500 nM T37848 C4DH0A 50938549 IC50 > 20000 nM T37848 CJ43IF 50941460 IC50 > 25000 nM T37848 CLIK30 50941729 IC50 > 10000 nM T37848 CP7B9V 50942696 IC50 = 2000 nM T37848 CX8N4D 50990920 IC50 > 10 nM T37848 CI32TR 50992246 IC50 > 25000 nM T37848 C2SHO8 50993865 IC50 = 17100 nM T37848 CNBU93 50994740 IC50 > 10000 nM T37848 CH82SZ 51000500 IC50 > 30000 nM T37848 CX48AD 51002362 IC50 = 10000 nM T37848 CX6PZ9 51003130 IC50 = 80 nM T37848 CAZQ43 51003133 IC50 > 20000 nM T37848 C8VNM2 51003549 IC50 > 50000 nM T37848 CP6NI2 51030711 IC50 > 30000 nM T37848 C70OGS 51030984 IC50 > 30000 nM T37848 CX28ZP 51030985 IC50 > 30000 nM T37848 CXB2Q6 51031001 IC50 > 30000 nM T37848 CUG03K 51033838 IC50 > 10000 nM T37848 C7OB2X 51035721 IC50 > 25000 nM T37848 C08FGN 51039225 IC50 = 4416 nM T37848 CS14BH 51039226 IC50 = 1281 nM T37848 CR70XF 51039227 IC50 > 10000 nM T37848 CA14XO 51051122 IC50 = 2500 nM T37848 C1RP3V 51051125 IC50 = 1900 nM T37848 C96AQN 51346908 IC50 > 30000 nM T37848 CGW84J 51346919 IC50 > 50000 nM T37848 C3I7XR 51346964 IC50 > 10000 nM T37848 CD2YU8 51351496 IC50 = 12000 nM T37848 C2UG4W 51351504 IC50 = 20000 nM T37848 CAO41L 51351511 IC50 > 30000 nM T37848 CG3PR6 52912222 IC50 = 21000 nM T37848 C8K6CQ 52916803 IC50 > 30000 nM T37848 CJ86KR 52917690 IC50 > 20000 nM T37848 CICZ45 52918012 IC50 < 300 nM T37848 CAXJ10 52918120 IC50 > 3162.28 nM T37848 CRN19G 52918121 IC50 > 3162.28 nM T37848 CTJ28K 52918135 IC50 > 50000 nM T37848 CJD25G 52920263 IC50 = 16000 nM T37848 CX9VO4 52932634 IC50 = 2000 nM T37848 C7VN1E 52934039 IC50 = 12900 nM T37848 CQ7EZ1 52934040 IC50 = 2000 nM T37848 CNOH36 52935183 IC50 = 1500 nM T37848 C12GTQ 52937251 IC50 = 2000 nM T37848 CQJG83 52940639 IC50 = 2900 nM T37848 CRCP02 52940664 IC50 = 0.5 nM T37848 C10WZR 52940895 IC50 = 3300 nM T37848 C2RW5A 52940961 IC50 > 6000 nM T37848 CSXY62 52941059 IC50 = 17100 nM T37848 CQW15U 52941269 IC50 > 50000 nM T37848 C1YLX8 52941699 IC50 = 24000 nM T37848 C80UVC 52941838 IC50 = 3500 nM T37848 C1QY0T 52941879 IC50 = 0.3 nM T37848 C6NR7I 52942081 IC50 > 30000 nM T37848 C3BO1Z 52942119 IC50 = 8500 nM T37848 C34WMT 52942456 IC50 = 68000 nM T37848 CHN91J 52942848 IC50 < 100 nM T37848 CV2ZC7 52943092 IC50 > 30 nM T37848 C56LMY 52943113 IC50 = 5.5 nM T37848 C0F3LG 52943305 IC50 > 100000 nM T37848 C3TK2O 52943442 IC50 = 18600 nM T37848 CHD7O6 52943758 IC50 = 13400 nM T37848 CA1B4V 52944247 IC50 = 2100 nM T37848 CZG75M 52944293 IC50 > 30 nM T37848 CTI28E 52944579 IC50 > 50000 nM T37848 CX0YD9 52944600 IC50 = 26600 nM T37848 CXTM57 52944645 IC50 > 30000 nM T37848 C4I6ML 52944843 IC50 = 7700 nM T37848 CT6SQ3 52944941 IC50 = 10200 nM T37848 C0OAD3 52945528 IC50 = 23.8 nM T37848 CQI9O0 52946720 IC50 = 1.5 nM T37848 CC29GI 52946733 IC50 > 30 nM T37848 CDW67R 52946750 IC50 = 7.1 nM T37848 CC60YV 52946759 IC50 = 30 nM T37848 CC38HD 52946978 IC50 = 13.6 nM T37848 CO7ZR1 52947102 IC50 = 14200 nM T37848 C2YK4B 52947710 IC50 = 10300 nM T37848 CXQ02F 52947930 IC50 = 6.4 nM T37848 CB3NQ0 52948140 IC50 = 900 nM T37848 C56NDZ 52948169 IC50 = 4800 nM T37848 C4WYC5 52948180 IC50 = 0.5 nM T37848 C48JMX 52948255 IC50 > 50000 nM T37848 C7SAC6 52948857 IC50 < 50 nM T37848 C43KTX 52948925 IC50 = 7200 nM T37848 C4LVO6 52948971 IC50 = 9400 nM T37848 C0HA6F 52949188 IC50 > 25000 nM T37848 CR36JQ 53232414 IC50 = 5100 nM T37848 C3DTV5 53233133 IC50 > 10000 nM T37848 C2RCZ0 53235503 IC50 > 20000 nM T37848 CV7BK2 53236350 IC50 = 1100 nM T37848 CQM95X 53236589 IC50 = 1900 nM T37848 C9RIJ7 53237893 IC50 = 11000 nM T37848 C5ZT7N 53237897 IC50 = 6100 nM T37848 C4KRV8 53237899 IC50 = 8700 nM T37848 C0H6TR 53237903 IC50 = 4400 nM T37848 CIP64Q 53238125 IC50 = 5500 nM T37848 C2AUL9 53248760 IC50 > 50000 nM T37848 CP3J9M 53248845 IC50 > 50000 nM T37848 CQIY23 53248846 IC50 > 50000 nM T37848 C9MHR0 53248847 IC50 > 50000 nM T37848 CG3LA9 53248849 IC50 > 20000 nM T37848 C2YXJ6 53248885 IC50 > 30000 nM T37848 C6RD7G 53249084 IC50 > 10000 nM T37848 CT9V3I 53251325 IC50 = 13800 nM T37848 CL62UR 53257683 IC50 = 3100 nM T37848 CB0TF8 53260999 IC50 = 1100 nM T37848 CV05UK 53261152 IC50 = 7800 nM T37848 CD35QU 53308640 IC50 > 10000 nM T37848 C1F3PN 53308743 IC50 = 26 nM T37848 CRI92N 53311230 IC50 > 10000 nM T37848 CQ9HO5 53311701 IC50 = 250 nM T37848 CL78NK 53316823 IC50 > 25000 nM T37848 C1-MAY-02 53317017 IC50 > 50000 nM T37848 C1P9YQ 53317572 IC50 = 7300 nM T37848 C7IMH5 53317594 IC50 > 10000 nM T37848 CT56HN 53317595 IC50 = 1405 nM T37848 CK27PC 53317643 IC50 = 33000 nM T37848 CXV3W2 53317718 IC50 > 50000 nM T37848 CP14EK 53317957 IC50 > 50000 nM T37848 CL45CT 53318503 IC50 > 5000 nM T37848 CDCA26 53318560 IC50 > 10000 nM T37848 C5F1IR 53318745 IC50 = 5000 nM T37848 CD0H8Z 53318872 IC50 > 10000 nM T37848 C90DGH 53318873 IC50 = 4840 nM T37848 C9MJ6C 53318874 IC50 > 10000 nM T37848 CB09MA 53318910 IC50 > 10 nM T37848 CJ2D3F 53319267 IC50 > 25000 nM T37848 COJ82D 53319320 IC50 > 50000 nM T37848 CK2G3D 53319480 IC50 > 25000 nM T37848 CTA23R 53319654 IC50 = 23000 nM T37848 CP31IL 53319749 IC50 = 3400 nM T37848 CXY8A4 53319905 IC50 > 38000 nM T37848 C7T9FB 53320163 IC50 > 50000 nM T37848 CWV40O 53320177 IC50 > 10000 nM T37848 CY5PO1 53320189 IC50 > 10000 nM T37848 CXF1S4 53320328 IC50 = 20100 nM T37848 CB84NG 53320778 IC50 > 25000 nM T37848 C5HL4R 53321372 IC50 > 25000 nM T37848 C9JVY1 53321494 IC50 > 10000 nM T37848 CQ9PR5 53321511 IC50 > 5000 nM T37848 CW28NZ 53321512 IC50 > 10000 nM T37848 C4X3IS 53321979 IC50 > 25000 nM T37848 CLD82J 53322084 IC50 > 25000 nM T37848 CMH54U 53322279 IC50 > 50000 nM T37848 CA91KC 53322692 IC50 > 25000 nM T37848 C9JUC1 53322838 IC50 = 1826 nM T37848 CEH78Z 53322839 IC50 = 1535 nM T37848 C78CYN 53322959 IC50 > 10000 nM T37848 CR57HN 53323639 IC50 = 7600 nM T37848 C6HPO5 53323744 IC50 > 10000 nM T37848 CX54CT 53323813 IC50 > 25000 nM T37848 C01OZU 53324167 IC50 = 4783 nM T37848 C1VNZ9 53324198 IC50 < 0.1 nM T37848 CC08MY 53324265 IC50 = 49000 nM T37848 CC1ER2 53324598 IC50 > 30000 nM T37848 C3QNR2 53325463 IC50 > 25000 nM T37848 CZN8B4 53325581 IC50 > 25000 nM T37848 C1WJH5 53325600 IC50 = 2820 nM T37848 CZ1SE0 53325908 IC50 > 50000 nM T37848 C1N7XO 53325966 IC50 > 25000 nM T37848 C28HNA 53326213 IC50 = 7700 nM T37848 C4VG5W 53326249 IC50 = 99500 nM T37848 CVNH56 53326712 IC50 = 4038 nM T37848 C4ZUJ9 53326724 IC50 > 10000 nM T37848 CU05TQ 53326725 IC50 = 3871 nM T37848 C9Z3WY 53326726 IC50 = 2751 nM T37848 CE9NR7 53326727 IC50 > 10000 nM T37848 C18TPG 53326909 IC50 > 25000 nM T37848 C7J8ZY 53327611 IC50 > 30000 nM T37848 C8PJ6E 53354789 IC50 = 9000 nM T37848 CYMP74 53354793 IC50 = 40000 nM T37848 C8ZRE3 53356518 IC50 = 9800 nM T37848 CUC1N3 53356519 IC50 > 17000 nM T37848 CL89US 53359023 IC50 > 50000 nM T37848 CRZL59 53361076 IC50 > 40000 nM T37848 C9H5YE 53361128 IC50 = 12000 nM T37848 CC7DZ4 53362086 IC50 > 50000 nM T37848 CX83CK 53362097 IC50 > 8900 nM T37848 C1F8IK 53363810 IC50 > 30000 nM T37848 C9GYZ3 53372790 IC50 = 4500 nM T37848 CT6K2O 53373472 IC50 = 6000 nM T37848 CL37YO 53380288 IC50 > 10000 nM T37848 C1Q0OJ 53382545 IC50 > 30000 nM T37848 C8NA4L 53384644 IC50 = 550 nM T37848 C19HFO 53386426 IC50 = 8900 nM T37848 CZWO31 53387025 IC50 > 100000 nM T37848 C7KM5B 53388319 IC50 = 40 nM T37848 CIGM78 53389570 IC50 > 30000 nM T37848 C64TJO 53391717 IC50 = 2650 nM T37848 C3Q6IL 53391718 IC50 = 10700 nM T37848 C6AYE3 53392451 IC50 > 100000 nM T37848 C47VGW 53393916 IC50 = 17600 nM T37848 C24FQU 53465297 IC50 > 12000 nM T37848 C0T5VA 53467975 IC50 > 11000 nM T37848 C2XHO3 53468206 IC50 > 11000 nM T37848 CX0R1K 53469059 IC50 = 19700 nM T37848 CV7C0D 53469060 IC50 = 7400 nM T37848 CCKD45 53469061 IC50 = 20500 nM T37848 C3SRN7 53469411 IC50 = 490 nM T37848 CK1C9O 53472113 IC50 = 19000 nM T37848 CE74YF 53473135 IC50 = 14000 nM T37848 C3SF8E 53473137 IC50 = 11000 nM T37848 CPN3C9 53473138 IC50 = 1500 nM T37848 CQNO62 53473139 IC50 > 30000 nM T37848 C8L2MJ 53473230 IC50 = 6000 nM T37848 CN1W0A 53473231 IC50 = 7000 nM T37848 CY1DW7 53473232 IC50 = 8000 nM T37848 CNS4A7 53473233 IC50 = 21000 nM T37848 CCN3Q2 53473234 IC50 > 30000 nM T37848 CL7D1V 53473235 IC50 = 3000 nM T37848 CZ8DA1 53473321 IC50 = 5000 nM T37848 CU7OV5 53473322 IC50 = 1000 nM T37848 C1HPT4 53473324 IC50 = 9000 nM T37848 CUN1Z2 53473393 IC50 = 12000 nM T37848 CE0I2P 53473394 IC50 > 30000 nM T37848 CW3Q5H 53473396 IC50 = 2000 nM T37848 CY0WF5 53473397 IC50 = 4000 nM T37848 C79FHR 53473483 IC50 = 600 nM T37848 CS87DG 53473484 IC50 = 7000 nM T37848 CITN21 53475321 IC50 > 20000 nM T37848 C9EF7S 53482945 IC50 > 100000 nM T37848 CFU8T7 53483937 IC50 > 30000 nM T37848 CG3FA9 53492750 IC50 = 15300 nM T37848 C4U5IX 53493001 IC50 > 35000 nM T37848 CL7K5O 53494954 IC50 = 3900 nM T37848 CE9K7U 53494972 IC50 > 10000 nM T37848 C7TR2W 53497131 IC50 > 30000 nM T37848 CS2RW9 53497480 IC50 = 16000 nM T37848 CSQ1Z3 53497481 IC50 > 60000 nM T37848 CN5HV2 53497485 IC50 = 53000 nM T37848 CGSN74 53497490 IC50 = 50000 nM T37848 C6NOA7 53497561 IC50 = 28000 nM T37848 CAE25J 53763992 IC50 = 158 nM T37848 CVA4I0 54576291 IC50 > 10000 nM T37848 CSAV94 54576503 IC50 > 10000 nM T37848 COF6B0 54577892 IC50 = 9400 nM T37848 C2ECL9 54577896 IC50 = 14600 nM T37848 CP24ZC 54579002 IC50 > 20000 nM T37848 CS1LM9 54580054 IC50 = 1000 nM T37848 C7FXV6 54580144 IC50 = 36000 nM T37848 CMDO43 54580283 IC50 = 21600 nM T37848 CQKX72 54580341 IC50 > 10000 nM T37848 C60LIJ 54580449 IC50 > 10000 nM T37848 C1NO3C 54580680 Ki = 240 nM T37848 CRB0W3 54580721 IC50 = 37000 nM T37848 C8PE1G 54581030 IC50 > 10000 nM T37848 C8S1LG 54581286 IC50 = 1600 nM T37848 C2XV8F 54581365 IC50 < 100 nM T37848 CQ0YA3 54581861 IC50 > 20000 nM T37848 CP2F1B 54582075 IC50 > 10000 nM T37848 CZNU23 54582076 IC50 > 10000 nM T37848 CSTG96 54582078 IC50 > 10000 nM T37848 C8V9GW 54582428 IC50 = 5200 nM T37848 C6N0BC 54582680 Ki = 130 nM T37848 CB8JV7 54582823 IC50 > 20000 nM T37848 CH6Q2Z 54583016 IC50 > 10000 nM T37848 C7LHV1 54583409 IC50 = 5500 nM T37848 CE5X6H 54583545 IC50 = 1075 nM T37848 C2RJM1 54583706 IC50 > 50000 nM T37848 CHP62C 54584119 IC50 = 10000 nM T37848 CY80OU 54584273 IC50 > 50000 nM T37848 CAO9B4 54584364 IC50 > 10000 nM T37848 CH95WP 54584618 Ki = 310 nM T37848 C37TZQ 54584868 IC50 > 30000 nM T37848 CAK7Z9 54585325 IC50 = 3300 nM T37848 CS51ZD 54585326 IC50 = 6700 nM T37848 CJIV69 54585540 IC50 > 30000 nM T37848 CI5W2A 54585926 IC50 = 1900 nM T37848 CSV1M4 54586281 IC50 > 10000 nM T37848 C01JOU 54586320 IC50 > 10000 nM T37848 C9FBH0 54586321 IC50 > 10000 nM T37848 CQ0G6R 54586630 IC50 = 8700 nM T37848 CQWI92 54586805 IC50 > 30000 nM T37848 CM0OQ3 54586893 IC50 > 10000 nM T37848 CK1NS7 54586894 IC50 > 10000 nM T37848 C6VQT3 54587171 IC50 = 2400 nM T37848 CO19MR 54587173 IC50 > 50000 nM T37848 C0VM3Y 54587553 IC50 = 2200 nM T37848 C5IAJ1 54587576 Ki = 250 nM T37848 C8MH6B 54587759 IC50 > 20000 nM T37848 CI9B8P 54670034 IC50 = 12589.25 nM T37848 CQ2EJ5 54670128 IC50 = 3162.28 nM T37848 C8JA6I 54670129 IC50 > 50118.72 nM T37848 C6J7OF 54670130 IC50 = 12589.25 nM T37848 C6W9QG 54671061 IC50 = 1584.89 nM T37848 CXU62W 54677935 IC50 > 40000 nM T37848 C0ZG2V 54709839 IC50 > 100000 nM T37848 CO75TL 54712015 IC50 > 50000 nM T37848 CLT3Q8 54716246 IC50 > 100000 nM T37848 C28RDF 54746913 IC50 > 50000 nM T37848 CMN1C6 54752118 IC50 > 10000 nM T37848 CZY7F9 54752621 IC50 > 7000 nM T37848 C69EQM 54752774 IC50 > 10000 nM T37848 CD8YN4 54753626 IC50 > 30000 nM T37848 CL32AY 54753627 IC50 > 30000 nM T37848 CBO2L1 54761157 IC50 > 40000 nM T37848 C0Y9ZG 54761473 IC50 > 10000 nM T37848 CS23GM 54762055 IC50 > 40000 nM T37848 CPS5V6 54764158 IC50 > 30000 nM T37848 CU62DN 54764919 IC50 > 30000 nM T37848 C4XCO3 54765024 IC50 = 140 nM T37848 C0T3KY 54765285 IC50 > 11000 nM T37848 CJ9B4P 54768039 IC50 > 10000 nM T37848 C79DVG 56589615 IC50 > 30000 nM T37848 C4S1HX 56589672 IC50 > 50000 nM T37848 C23NQS 56593147 IC50 > 20000 nM T37848 CXSQ19 56593712 IC50 = 74800 nM T37848 C4U6BD 56593857 IC50 > 100000 nM T37848 CHD79F 56594864 IC50 = 1100 nM T37848 CMQ2J3 56594865 IC50 = 2500 nM T37848 C6FE3Z 56594866 IC50 = 1000 nM T37848 CS3E5I 56594867 IC50 < 100 nM T37848 C91PGO 56603115 IC50 > 50000 nM T37848 C5ES6P 56603116 IC50 = 6400 nM T37848 CVI51O 56603118 IC50 > 50000 nM T37848 C2IM6T 56603174 IC50 > 50000 nM T37848 CH05TN 56603175 IC50 > 50000 nM T37848 CDL94H 56603301 IC50 = 13300 nM T37848 C9D1MV 56603353 IC50 > 50000 nM T37848 C9ZF6B 56643412 IC50 > 25000 nM T37848 C4N0WL 56645363 IC50 > 50000 nM T37848 C57NSZ 56645568 IC50 > 50000 nM T37848 C6PUX9 56645570 IC50 > 50000 nM T37848 CTW6K2 56645571 IC50 = 8235 nM T37848 CBJ4V8 56649677 IC50 = 9000 nM T37848 C5OT6W 56658248 Ki = 0.022 nM T37848 CPJ7D3 56658546 IC50 > 30000 nM T37848 C7AG6I 56658547 IC50 > 30000 nM T37848 C6W5UT 56658548 IC50 > 30000 nM T37848 CFT9V8 56659147 IC50 > 25000 nM T37848 CGID30 56659201 IC50 > 10000 nM T37848 CX31TJ 56661748 Ki = 0.026 nM T37848 C2QTH5 56662000 IC50 > 30000 nM T37848 CC1GK4 56665357 IC50 > 30000 nM T37848 CU4J0H 56668366 IC50 = 9300 nM T37848 CC9XR7 56669562 IC50 > 10000 nM T37848 CXE9A8 56669563 IC50 > 8000 nM T37848 C9MW0X 56670034 IC50 < 10000 nM T37848 CK9L4C 56672570 IC50 > 30000 nM T37848 C1E4CX 56673467 IC50 > 50000 nM T37848 CADI17 56673550 IC50 = 1000 nM T37848 C58RPD 56675666 IC50 = 26 nM T37848 CKVS08 56676902 IC50 = 470 nM T37848 CZP86D 56677285 IC50 > 30000 nM T37848 C7QW5F 56678507 IC50 = 6800 nM T37848 CW7QF9 56679101 IC50 > 30000 nM T37848 CUIB93 56679632 IC50 = 51900 nM T37848 CBOK07 56682298 IC50 = 20 nM T37848 CK73UC 56683046 IC50 > 6000 nM T37848 CR0E4M 56683440 IC50 > 50000 nM T37848 CJC19B 56683709 IC50 > 30000 nM T37848 CY3G8F 56834936 IC50 = 24000 nM T37848 CPN57V 56834986 IC50 > 10000 nM T37848 CR7LS4 56835090 IC50 > 30000 nM T37848 C70GHX 56835991 IC50 > 50000 nM T37848 CK7HJ8 56837192 IC50 = 2600 nM T37848 CH2AY6 56838673 IC50 > 30000 nM T37848 C3OE8N 56838888 IC50 > 30000 nM T37848 CBHT83 56840376 IC50 = 5000 nM T37848 CVYF04 56840671 IC50 > 10000 nM T37848 CR8KU2 56840672 IC50 > 10000 nM T37848 CKY51C 56847605 IC50 = 54000 nM T37848 CUY28J 56850524 IC50 = 8.5 nM T37848 CK0I6Q 56850525 IC50 = 5.5 nM T37848 C1U7XJ 56924869 IC50 > 30000 nM T37848 CDVO63 56928630 IC50 = 12000 nM T37848 CZRQ14 56929159 IC50 = 54000 nM T37848 C9IVD0 56929216 IC50 > 10000 nM T37848 C90URY 56929249 IC50 = 54000 nM T37848 CZ25SN 56935695 IC50 > 10000 nM T37848 C9KI7Q 56940718 IC50 = 50 nM T37848 CPAU51 56943206 IC50 > 10000 nM T37848 CR2O1Z 56946068 Ki = 800 nM T37848 CI3X1S 56946069 Ki = 32900 nM T37848 C5CXM7 56946070 Ki = 20100 nM T37848 CRVI60 56946173 Ki = 15930 nM T37848 C1FPQ0 56946174 Ki = 6900 nM T37848 CE71VQ 56946175 Ki = 2700 nM T37848 CC3VZ7 56946176 Ki = 2200 nM T37848 CG72VK 56946177 Ki = 8400 nM T37848 C9EM3S 56946178 Ki = 2200 nM T37848 CHK14G 56946281 Ki = 3000 nM T37848 CI04WC 56948248 IC50 = 120 nM T37848 CL16UQ 56949326 IC50 = 9500 nM T37848 C71JRF 56949451 IC50 = 900 nM T37848 C89PEN 56949822 IC50 > 10000 nM T37848 C1K8TD 56949966 IC50 > 10000 nM T37848 C5LJE8 56951456 IC50 = 25800 nM T37848 C6N0ZI 56951457 IC50 > 27000 nM T37848 CL90EM 56951458 IC50 = 11800 nM T37848 CP6AS2 56952795 IC50 > 50000 nM T37848 CWB5H7 56953768 IC50 = 26300 nM T37848 CS0HF1 56953769 IC50 = 5330 nM T37848 CPJ7X3 56953770 IC50 = 15700 nM T37848 CK7M6W 56953771 IC50 = 50000 nM T37848 CO96BR 56953896 IC50 = 16400 nM T37848 CJ0WM6 56953897 IC50 = 6230 nM T37848 C4UV1D 56953898 IC50 = 8340 nM T37848 CPKI96 56954010 IC50 = 4910 nM T37848 C6Q8BZ 56954011 IC50 = 1870 nM T37848 C5G4UX 56954012 IC50 = 2810 nM T37848 C8UQ2S 56954013 IC50 = 2490 nM T37848 CHQA53 56954137 IC50 = 3560 nM T37848 CZGE53 56954138 IC50 = 10700 nM T37848 CGRC25 56954242 IC50 = 7146 nM T37848 CRT0Y2 56954243 IC50 = 301 nM T37848 CAK91L 56955954 IC50 > 20000 nM T37848 CD3SZ1 56959836 IC50 > 1000 nM T37848 CN2GI7 56959991 IC50 = 1600 nM T37848 C1TR4E 56963091 IC50 = 33000 nM T37848 CKN0Z8 56964577 IC50 > 25000 nM T37848 CS7U9L 56965952 IC50 > 10000 nM T37848 C1K2YU 56968076 IC50 = 57000 nM T37848 CT67IO 57325589 IC50 > 25000 nM T37848 CV5CP4 57326678 IC50 = 5500 nM T37848 CQT5I3 57328465 IC50 > 27000 nM T37848 CY58ZD 57330086 IC50 = 1100 nM T37848 CW8B4D 57330208 IC50 > 27000 nM T37848 C4D1LZ 57330959 IC50 = 18000 nM T37848 CLB5K0 57331386 IC50 > 10000 nM T37848 CGUA26 57331668 IC50 > 50000 nM T37848 C8C1EW 57334262 IC50 = 7900 nM T37848 CU5BD9 57336812 IC50 = 11000 nM T37848 CFW0D1 57339435 IC50 = 13000 nM T37848 CL45WN 57345320 IC50 > 12000 nM T37848 C8CGX9 57345520 IC50 = 700 nM T37848 CT8VZ6 57345658 IC50 > 30000 nM T37848 C7O0AI 57345659 IC50 > 30000 nM T37848 C3L9ZA 57345660 IC50 > 30000 nM T37848 CZK3M1 57345661 IC50 > 30000 nM T37848 C34DJP 57384236 IC50 > 50000 nM T37848 CEOC15 57384237 IC50 > 50000 nM T37848 CY50WC 57384238 IC50 > 50000 nM T37848 C7S0ZR 57384239 IC50 = 18000 nM T37848 C9Q4VL 57384270 IC50 = 2100 nM T37848 CDS03B 57384271 IC50 = 800 nM T37848 CBKI24 57384272 IC50 = 9200 nM T37848 C6IAW5 57384273 IC50 = 6700 nM T37848 C42JEK 57384274 IC50 = 400 nM T37848 C2XN1G 57384481 IC50 > 50000 nM T37848 CR73IZ 57384482 IC50 > 50000 nM T37848 CR2M5H 57384483 IC50 > 50000 nM T37848 CQ72HI 57384749 IC50 > 50000 nM T37848 C68KGE 57384750 IC50 > 50000 nM T37848 CCT5D4 57386783 IC50 > 50000 nM T37848 CC30XZ 57386784 IC50 > 50000 nM T37848 C79BXP 57386785 IC50 > 50000 nM T37848 CM6DV7 57387028 IC50 > 50000 nM T37848 C0GS4F 57387282 IC50 > 50000 nM T37848 C0TL9C 57387283 IC50 > 50000 nM T37848 CRV2P5 57387539 IC50 > 50000 nM T37848 CAU3G9 57387540 IC50 > 50000 nM T37848 CL2AO8 57387541 IC50 > 50000 nM T37848 C0XWL8 57387542 IC50 > 50000 nM T37848 CC4DK0 57387775 IC50 > 50000 nM T37848 CZ0W8T 57387809 IC50 = 300 nM T37848 CJA0T7 57388041 IC50 = 400 nM T37848 C6ATQ0 57390715 IC50 = 3200 nM T37848 CP8D5L 57390807 IC50 = 5600 nM T37848 CDJC72 57390808 IC50 = 13000 nM T37848 CE03ZS 57390809 IC50 = 8900 nM T37848 CWR4E5 57390923 IC50 > 17000 nM T37848 C0RAD8 57390924 IC50 > 17000 nM T37848 C5OJP0 57391102 IC50 > 25000 nM T37848 CD07RK 57391165 IC50 = 12900 nM T37848 CC76GU 57391166 IC50 = 12200 nM T37848 CR8MW2 57391205 IC50 > 10000 nM T37848 C2AR3V 57391609 IC50 <= 3000 nM T37848 CKPB03 57391802 IC50 <= 3000 nM T37848 C8SW9E 57391803 IC50 <= 3000 nM T37848 C5UWC6 57391804 IC50 <= 3000 nM T37848 C78QEY 57391805 IC50 <= 3000 nM T37848 C95QGI 57391832 IC50 = 11 nM T37848 C48NQU 57391833 IC50 = 220 nM T37848 CT2R0D 57391834 IC50 = 280 nM T37848 C2D9AX 57391850 IC50 = 710 nM T37848 C2RF6A 57391851 IC50 = 480 nM T37848 CXB7E6 57391852 IC50 = 1200 nM T37848 CBWK43 57391853 IC50 = 290 nM T37848 CT96ZS 57392011 IC50 = 900 nM T37848 C16PSG 57392623 IC50 = 6000 nM T37848 CFM8E5 57392624 IC50 = 2200 nM T37848 C4QYJ6 57392724 IC50 > 17000 nM T37848 C9OLQ7 57392788 IC50 > 20000 nM T37848 C9JYK4 57392932 IC50 = 20000 nM T37848 CNQ9B2 57392969 IC50 > 10000 nM T37848 CAV09E 57393151 IC50 > 172000 nM T37848 CF94AV 57393565 IC50 = 30 nM T37848 CHU04N 57393566 IC50 = 5300 nM T37848 CSQ64Y 57393587 IC50 = 61 nM T37848 CJE25R 57393588 IC50 = 200 nM T37848 CB6JG7 57393589 IC50 = 44 nM T37848 C6JCU0 57393590 IC50 = 4600 nM T37848 CHA2Q7 57394339 IC50 = 5000 nM T37848 CS8M9I 57394340 IC50 = 1600 nM T37848 CLP4Z8 57394341 IC50 = 3600 nM T37848 C8PWV4 57394342 IC50 = 3500 nM T37848 C16OJD 57394343 IC50 = 6000 nM T37848 C0AJM8 57394344 IC50 = 31000 nM T37848 C6HR3Q 57394345 IC50 = 2800 nM T37848 CWDY79 57394441 IC50 > 17000 nM T37848 CCEO27 57394520 IC50 = 3300 nM T37848 C04IST 57394707 IC50 > 10000 nM T37848 CNOH63 57394711 IC50 > 10000 nM T37848 C5USX7 57395248 IC50 <= 3000 nM T37848 CJ80BU 57395249 IC50 <= 3000 nM T37848 CTDA90 57395276 IC50 = 1700 nM T37848 CA03VI 57395277 IC50 = 360 nM T37848 CSO4Z0 57395278 IC50 = 4700 nM T37848 CB09IO 57395287 IC50 > 20000 nM T37848 CA32IO 57395298 IC50 = 26 nM T37848 CNC0G9 57395299 IC50 = 90 nM T37848 CQS1Y0 57395300 IC50 = 47 nM T37848 C3EQP0 57395301 IC50 = 79 nM T37848 CF67DY 57395302 IC50 = 14000 nM T37848 CHX4Z7 57396095 IC50 = 7200 nM T37848 CRS39Y 57396096 IC50 = 2300 nM T37848 CLEH95 57396097 IC50 = 9300 nM T37848 C4NVE2 57396098 IC50 = 5800 nM T37848 C7PT9Q 57396099 IC50 = 2000 nM T37848 C23WQH 57396100 IC50 = 2400 nM T37848 C8KMS2 57396206 IC50 > 17000 nM T37848 CE75UA 57396432 IC50 < 200 nM T37848 C9K7YS 57396433 IC50 = 7100 nM T37848 CWE8N9 57396434 IC50 = 300 nM T37848 C6HBG0 57396813 IC50 > 5900 nM T37848 CB71KN 57396814 IC50 = 1200 nM T37848 C0P8KM 57397016 IC50 <= 3000 nM T37848 CE85SV 57397017 IC50 >= 10000 nM T37848 CBHJ53 57397047 IC50 = 200 nM T37848 C25FTZ 57397056 IC50 = 15600 nM T37848 CDR0K6 57397067 IC50 = 82 nM T37848 CTBP48 57397068 IC50 = 98 nM T37848 CBRN40 57397069 IC50 = 2900 nM T37848 CU4FW8 57397383 IC50 > 25000 nM T37848 CH32BO 57397434 IC50 < 200 nM T37848 CQS0M5 57397654 IC50 > 30000 nM T37848 CD7M5V 57397795 IC50 = 6900 nM T37848 CH4Z3O 57397916 IC50 = 1100 nM T37848 CW97SN 57398006 IC50 > 17000 nM T37848 C65DMS 57398065 IC50 = 7200 nM T37848 CCS9O0 57398066 IC50 > 20000 nM T37848 CDWI58 57398224 IC50 = 1000 nM T37848 CDSH51 57398573 IC50 = 7800 nM T37848 C7WH5G 57398574 IC50 < 200 nM T37848 CSU2O9 57398779 IC50 <= 3000 nM T37848 C4DM3N 57398809 IC50 = 130 nM T37848 CF13IE 57398846 IC50 = 1500 nM T37848 C32IVG 57398848 IC50 = 70 nM T37848 CB42RN 57399556 IC50 = 1600 nM T37848 C01KCU 57399665 IC50 > 17000 nM T37848 CYC7S5 57399874 IC50 = 300 nM T37848 C2GO5M 57400235 IC50 = 4600 nM T37848 CDQ57A 57400458 IC50 <= 3000 nM T37848 CED9C4 57400459 IC50 <= 3000 nM T37848 C1A6CD 57400491 IC50 = 270 nM T37848 CE82XL 57400502 IC50 = 4900 nM T37848 CWZ50O 57400503 IC50 = 9500 nM T37848 C5MG6Q 57400504 IC50 = 10600 nM T37848 CJBU02 57400505 IC50 = 5800 nM T37848 C8JR5T 57400522 IC50 = 310 nM T37848 CML28J 57400523 IC50 = 110 nM T37848 C3D0SL 57400524 IC50 = 60 nM T37848 CUYK04 57401306 IC50 = 6400 nM T37848 CSQK78 57401307 IC50 = 1900 nM T37848 C8GC4D 57401308 IC50 = 15000 nM T37848 CFL71K 57401309 IC50 = 700 nM T37848 CYX43T 57401419 IC50 > 17000 nM T37848 CMS98N 57402038 IC50 = 600 nM T37848 C0MKN9 57402230 IC50 = 15800 nM T37848 CV2ME6 57402260 IC50 <= 3000 nM T37848 CW94QA 57402262 IC50 <= 3000 nM T37848 CMJA69 57402263 IC50 >= 10000 nM T37848 CT48QS 57402295 IC50 = 48 nM T37848 CXT2L1 57402315 IC50 > 20000 nM T37848 C1HN8Y 57402329 IC50 = 210 nM T37848 CY45EB 57402330 IC50 = 600 nM T37848 CY97BO 57402969 IC50 = 7800 nM T37848 CQ1ZV2 57403067 IC50 = 5600 nM T37848 C1T0AD 57403169 IC50 > 17000 nM T37848 C12QCM 57403170 IC50 > 17000 nM T37848 CX94UQ 57403171 IC50 = 7000 nM T37848 CSL60R 57403230 IC50 = 11000 nM T37848 C78GME 57403231 IC50 = 5400 nM T37848 CU5J8W 57403232 IC50 = 9000 nM T37848 CKVH81 57403233 IC50 > 20000 nM T37848 C6B3IK 57403377 IC50 = 300 nM T37848 CW54GL 57403378 IC50 = 1100 nM T37848 CI9A1D 57403379 IC50 > 20000 nM T37848 C4EWA9 57403779 IC50 = 2900 nM T37848 C1H5LA 57403780 IC50 < 200 nM T37848 C4RHF3 57404027 IC50 > 30000 nM T37848 CU8PE6 57404044 IC50 = 92 nM T37848 C40WQO 57404045 IC50 = 55 nM T37848 C1MOD0 57404046 IC50 = 53 nM T37848 CTJI57 57404047 IC50 = 560 nM T37848 CI1A8M 57404048 IC50 = 22000 nM T37848 CPGR16 57404049 IC50 = 26000 nM T37848 CKU6E8 57404500 IC50 > 30000 nM T37848 C6XA7G 57405264 IC50 > 30000 nM T37848 CED47A 57410062 IC50 = 40000 nM T37848 CUOV05 57411066 IC50 > 30000 nM T37848 C1BVX6 57411134 IC50 = 40000 nM T37848 CD0W2I 57411254 IC50 = 40000 nM T37848 C6U4LO 57411256 IC50 = 40000 nM T37848 CC5DO3 57411369 IC50 = 40000 nM T37848 C56RBS 57411372 IC50 = 40000 nM T37848 CK5QX7 57411488 IC50 = 40000 nM T37848 C90LNK 57411715 IC50 = 40000 nM T37848 CPXE40 57411716 IC50 = 40000 nM T37848 CE6RY5 57411836 IC50 = 40 nM T37848 C5JOX3 57411837 IC50 = 40000 nM T37848 CDMI53 57415260 IC50 = 130 nM T37848 C6GWV8 57415261 IC50 = 3400 nM T37848 CE63TG 57415391 IC50 = 280 nM T37848 COUZ63 57494822 IC50 = 737 nM T37848 C72OWZ 57502386 IC50 = 200 nM T37848 C9Z6QJ 57502388 IC50 = 24000 nM T37848 C37SMZ 57505249 IC50 > 100000 nM T37848 CUG89V 57506726 IC50 = 510 nM T37848 CVOP28 57506727 IC50 = 600 nM T37848 C48BYL 57506732 IC50 < 100 nM T37848 CBZS07 57506734 IC50 = 9100 nM T37848 CFH0J4 57506741 IC50 > 10000 nM T37848 CI30AW 57506743 IC50 > 10000 nM T37848 CL47BS 57506744 IC50 > 10000 nM T37848 C23FTC 57510027 IC50 > 20000 nM T37848 C7I4QD 57519510 IC50 > 50000 nM T37848 C3N4MF 57520842 IC50 > 50000 nM T37848 CEL56T 57520942 IC50 > 50000 nM T37848 CBC85H 57522018 IC50 = 1030 nM T37848 CIK6G9 57522019 IC50 < 200 nM T37848 CW23VX 57522130 IC50 = 400 nM T37848 CT13YK 57522131 IC50 = 1530 nM T37848 C20IFP 57522132 IC50 = 7800 nM T37848 CW50IU 57522133 IC50 = 1300 nM T37848 C6E5BW 57522134 IC50 = 8000 nM T37848 C43URP 57522135 IC50 = 420 nM T37848 CYU9J7 57522248 IC50 = 430 nM T37848 CWLD45 57522249 IC50 = 600 nM T37848 C2K5MR 57522250 IC50 = 2400 nM T37848 C6HTG0 57522251 IC50 = 2900 nM T37848 C1HRZ7 57544434 IC50 = 3100 nM T37848 CN0CF4 57544848 IC50 = 2910 nM T37848 CAQ71K 57574919 IC50 > 20000 nM T37848 CASM07 57574933 IC50 = 17200 nM T37848 CM1EK8 57574953 IC50 = 15400 nM T37848 CX4F6L 57574973 IC50 = 13800 nM T37848 CY5D1K 57574980 IC50 = 1900 nM T37848 C9CD2Y 57574990 IC50 = 7700 nM T37848 C3XGL6 57574995 IC50 > 20000 nM T37848 CR7K1C 57575007 IC50 = 4000 nM T37848 CG93BU 57575012 IC50 = 6100 nM T37848 CPE25J 57575026 IC50 = 3300 nM T37848 C1EC2O 57576905 IC50 = 150 nM T37848 CWUR92 57577004 IC50 = 10000 nM T37848 C8JQT0 57633016 IC50 = 3700 nM T37848 CKH8C1 57633047 IC50 = 2300 nM T37848 CSV52O 57633056 IC50 = 4900 nM T37848 CV6J8N 57633096 IC50 = 5900 nM T37848 C25KIP 57633210 IC50 = 3600 nM T37848 CB30PQ 57656715 IC50 = 1600 nM T37848 CV2J9A 57663655 IC50 = 64000 nM T37848 CP2B1Q 57686448 IC50 = 2000000 nM T37848 CTM6K5 57690900 IC50 = 22000 nM T37848 C35GXV 57720515 EC50 = 9000 nM T37848 C58TKU 57773771 IC50 = 270 nM T37848 C0JCN7 57798480 IC50 > 50000 nM T37848 CF94GH 57812483 IC50 > 20000 nM T37848 C2BR4G 57812601 IC50 = 1600 nM T37848 C9OBT1 57869953 IC50 > 50000 nM T37848 C7C4VE 57870158 IC50 > 50000 nM T37848 C2CR3O 57870171 IC50 > 50000 nM T37848 C0QFL3 57877765 IC50 > 50000 nM T37848 CG23VP 57941404 IC50 = 22600 nM T37848 C6C8UT 57941522 IC50 > 50000 nM T37848 CY4O6Z 57965013 IC50 = 1800 nM T37848 CP28UL 57965039 IC50 > 25000 nM T37848 CANZ90 57994936 IC50 > 20000 nM T37848 C8NW0C 58017500 IC50 = 28000 nM T37848 C67MSZ 58017509 IC50 = 1200 nM T37848 CG9V4E 58017514 IC50 = 1800 nM T37848 C7M3DS 58017531 IC50 > 20000 nM T37848 CW1SD9 58017538 IC50 > 50000 nM T37848 CJ6Y1B 58026134 IC50 > 30000 nM T37848 CV1RX3 58026153 IC50 = 2000 nM T37848 C19XQV 58026164 IC50 = 10 nM T37848 CR7H3O 58026170 IC50 > 30000 nM T37848 C7XL3D 58026176 IC50 = 3000 nM T37848 CY9CA0 58031728 IC50 = 1000 nM T37848 C3J7XM 58063084 IC50 = 6700 nM T37848 C1EVX0 58063117 IC50 = 5800 nM T37848 CGBY54 58063225 IC50 > 10000 nM T37848 C0P8VW 58063334 IC50 > 10000 nM T37848 CZO2J1 58063487 IC50 > 10000 nM T37848 C5B0RJ 58083331 IC50 > 50000 nM T37848 C1C6OS 58083336 IC50 = 29000 nM T37848 C6DZ0X 58083358 IC50 = 45000 nM T37848 CSC1K6 58109236 IC50 > 50000 nM T37848 CS05MK 58109240 IC50 > 50000 nM T37848 CDC28F 58109250 IC50 > 50000 nM T37848 CY5V0J 58109251 IC50 = 2100 nM T37848 C4E2RC 58109371 IC50 = 12700 nM T37848 C2EY8P 58109378 IC50 = 27000 nM T37848 C05LAK 58109398 IC50 > 30000 nM T37848 CJ07OW 58109450 IC50 > 30000 nM T37848 C5JGU1 58109561 IC50 > 30000 nM T37848 CZAJ57 58109626 IC50 > 30000 nM T37848 CZY78L 58109663 IC50 = 6600 nM T37848 C4SC0Z 58109674 IC50 > 50000 nM T37848 CTQ2N4 58109704 IC50 = 23000 nM T37848 CRZU03 58109712 IC50 > 30000 nM T37848 C4NJG2 58109725 IC50 = 10000 nM T37848 C1EF0B 58109729 IC50 > 50000 nM T37848 C2QB4E 58143638 IC50 = 7900 nM T37848 C3GKN6 58143653 IC50 = 2900 nM T37848 C53ESG 58143660 IC50 = 500 nM T37848 CWXC70 58180596 IC50 = 3000 nM T37848 CBZX94 58199027 IC50 > 30000 nM T37848 CB72QI 58204997 IC50 > 10000 nM T37848 C93STQ 58239274 IC50 = 15000 nM T37848 C2SE1Z 58239287 IC50 > 20000 nM T37848 CI45ZP 58269513 IC50 > 30000 nM T37848 CK10DA 58269516 IC50 = 6000 nM T37848 CV9FC4 58269518 IC50 > 30000 nM T37848 CM1GN4 58269523 IC50 = 24000 nM T37848 CAY0H7 58269562 IC50 > 30000 nM T37848 CN13SI 58269563 IC50 = 15000 nM T37848 CPQ0Z4 58269588 IC50 > 30000 nM T37848 C8A3JQ 58269598 IC50 = 400 nM T37848 CD18IU 58269609 IC50 = 22000 nM T37848 CQV75S 58269620 IC50 = 24500 nM T37848 C26OPT 58269625 IC50 > 30000 nM T37848 C8ILS3 58269629 IC50 = 13000 nM T37848 C5VFQ7 58269655 IC50 = 11000 nM T37848 CQ63WZ 58269663 IC50 = 3000 nM T37848 C2PYB1 58269668 IC50 = 26000 nM T37848 CI3P0D 58269670 IC50 > 30000 nM T37848 C5RF8T 58269685 IC50 > 30000 nM T37848 C4OS3J 58269689 IC50 > 30000 nM T37848 C3CFB8 58269691 IC50 = 26000 nM T37848 CJ4B6P 58299601 IC50 > 10000 nM T37848 CU24DE 58299617 IC50 > 10000 nM T37848 CT78UE 58299836 IC50 > 10000 nM T37848 C1I0OB 58299870 IC50 = 9500 nM T37848 CD87NL 58300031 IC50 > 10000 nM T37848 C5RB1P 58300060 IC50 > 10000 nM T37848 C63AEW 58300068 IC50 > 10000 nM T37848 CZA32V 58344912 IC50 > 10000 nM T37848 CPVF85 58344916 IC50 > 10000 nM T37848 CY62SG 58345029 IC50 > 10000 nM T37848 CMXC37 58365250 IC50 > 20000 nM T37848 C4EPA5 58365345 IC50 > 20000 nM T37848 CO53TZ 58365501 IC50 > 20000 nM T37848 CXY58G 58365527 IC50 > 20000 nM T37848 CON6K1 58365686 IC50 > 20000 nM T37848 CVP17Q 58365704 IC50 > 20000 nM T37848 CZ6X0Y 58365744 IC50 > 20000 nM T37848 CX8Y6Z 58365813 IC50 > 20000 nM T37848 C3WB9I 58365828 IC50 > 20000 nM T37848 C5CRB1 58365867 IC50 > 20000 nM T37848 CF6A8Y 58365941 IC50 > 20000 nM T37848 C35RYZ 58365945 IC50 > 20000 nM T37848 CJI25C 58365995 IC50 > 20000 nM T37848 C3QI6Y 58366053 IC50 > 20000 nM T37848 C6AC9L 58366064 IC50 > 20000 nM T37848 CC67BX 58366073 IC50 > 20000 nM T37848 C54QRX 58394136 IC50 > 50000 nM T37848 C0F3BO 58394783 IC50 > 10000 nM T37848 C0X7IK 58394837 IC50 = 7900 nM T37848 CASI81 58395078 IC50 = 8800 nM T37848 CWBM72 58395283 IC50 = 6700 nM T37848 CZL8H3 58437582 IC50 > 20000 nM T37848 C48NCZ 58437683 IC50 = 13200 nM T37848 CI0A7Z 58437687 IC50 > 20000 nM T37848 C0OBW7 58438170 IC50 = 5000 nM T37848 CS6L4E 58438199 IC50 = 9400 nM T37848 CSE71O 58438284 IC50 > 20000 nM T37848 C9UK7P 58438475 IC50 = 2500 nM T37848 C6BZ0G 58439416 IC50 = 18000 nM T37848 CWYK20 58485289 IC50 = 11000 nM T37848 CN2E9O 58485355 IC50 = 1800 nM T37848 CAW51G 58486138 IC50 = 2800 nM T37848 CRB42N 58486297 IC50 = 300 nM T37848 C35FWX 58486367 IC50 > 10000 nM T37848 CJV84Q 58534983 IC50 > 10000 nM T37848 C6JKM0 58834906 IC50 > 100000 nM T37848 CF9Z0L 58834953 IC50 > 26000 nM T37848 C4PWA9 58835024 IC50 > 40000 nM T37848 CCR4T7 58835217 IC50 > 73000 nM T37848 C5UJ4T 58863082 IC50 > 30000 nM T37848 CNM1V0 58863113 IC50 > 30000 nM T37848 C5FOK7 58863126 IC50 > 30000 nM T37848 CU89KE 58863146 IC50 = 22000 nM T37848 CNE1Q4 58863165 IC50 > 30000 nM T37848 CM58WY 58863171 IC50 = 30000 nM T37848 CO4NR9 58863217 IC50 > 30000 nM T37848 CK5P3B 58863232 IC50 > 30000 nM T37848 C6AY0Z 58864297 IC50 = 6900 nM T37848 C9ZE7J 58874273 IC50 > 50000 nM T37848 C7CE6L 58950132 IC50 = 21400 nM T37848 C6ZQ3C 58973420 IC50 = 610 nM T37848 CUH6F9 59122522 IC50 = 300 nM T37848 CCQM76 59153288 IC50 > 50000 nM T37848 CL9R5T 59156709 IC50 > 50000 nM T37848 C3L4JY 59176329 IC50 > 10000 nM T37848 CU4Y6H 59177057 IC50 = 830 nM T37848 C0U1HA 59179260 IC50 > 10000 nM T37848 CK7T6D 59179887 IC50 > 10000 nM T37848 C6DG2S 59190464 IC50 > 1000 nM T37848 CL9R5M 59190503 IC50 > 1000 nM T37848 CQHS47 59190547 IC50 = 398.11 nM T37848 C79GHB 59190548 IC50 > 1000 nM T37848 CI26UZ 59201574 IC50 = 7100 nM T37848 CDM57O 59239077 IC50 = 3300 nM T37848 CQ4HD1 59239114 IC50 = 900 nM T37848 C6MQA3 59239348 IC50 > 10000 nM T37848 C2BX0H 59239374 IC50 = 2500 nM T37848 CP64KI 59239424 IC50 = 8400 nM T37848 CJ6R8Q 59251679 IC50 > 25000 nM T37848 CGB6E7 59251838 IC50 = 50 nM T37848 C3UDA9 59251852 IC50 = 800 nM T37848 C2PJ4N 59271992 IC50 = 4000 nM T37848 CUE79I 59272004 IC50 = 4400 nM T37848 CZCV65 59272024 IC50 = 3100 nM T37848 C7AOL2 59272040 IC50 = 3200 nM T37848 CK8GF7 59272204 IC50 > 10000 nM T37848 CTQ42U 59272220 IC50 <= 200 nM T37848 C1MTZ2 59272228 IC50 = 6400 nM T37848 C0S6UA 59272254 IC50 <= 200 nM T37848 C2QBE7 59272265 IC50 > 10000 nM T37848 CKO4S7 59272298 IC50 = 10000 nM T37848 C9VNB7 59275242 IC50 = 4100 nM T37848 CD4S2Z 59275372 IC50 = 63 nM T37848 CTF1U6 59275404 IC50 > 13000 nM T37848 CI5E9M 59275443 IC50 = 2100 nM T37848 CYE54A 59275494 IC50 = 73 nM T37848 C4KU2S 59278286 IC50 = 17000 nM T37848 CEAY32 59278314 IC50 > 30000 nM T37848 CBWJ84 59291203 IC50 < 1000 nM T37848 C6A3KL 59293676 IC50 > 10000 nM T37848 CC14ZL 59293709 IC50 > 10000 nM T37848 C0R3TX 59293715 IC50 > 10000 nM T37848 CB2Z4R 59293755 IC50 > 10000 nM T37848 C8AL6C 59293763 IC50 > 10000 nM T37848 C19YVT 59377518 IC50 > 32000 nM T37848 C1JK7V 59377559 IC50 > 50000 nM T37848 CEB4Z6 59389144 IC50 < 400 nM T37848 C2XTM4 59389145 IC50 > 30000 nM T37848 C34OHS 59389193 IC50 < 300 nM T37848 CYJ43P 59389208 IC50 = 1900 nM T37848 C1U4XM 59389234 IC50 = 4300 nM T37848 CFDG19 59401765 IC50 > 30000 nM T37848 CC5QW1 59401793 IC50 > 30000 nM T37848 CNOI48 59401886 IC50 > 30000 nM T37848 CJ2Y3A 59414201 IC50 = 150 nM T37848 CD9U3W 59414209 IC50 = 100 nM T37848 CPUZ69 59447115 IC50 = 10000 nM T37848 CVZ09Q 59454159 IC50 = 3000 nM T37848 CK6LX0 59454220 IC50 = 4000 nM T37848 C2SDN1 59454252 IC50 = 21000 nM T37848 CK6W7I 59536635 IC50 > 10000 nM T37848 CA9NE4 59548712 IC50 > 30000 nM T37848 CM1G2P 59568656 IC50 > 50000 nM T37848 CJLD97 59603304 IC50 = 28 nM T37848 CYP12T 59603305 IC50 = 40 nM T37848 C1NW7Q 59603306 IC50 = 90 nM T37848 CJ0H1Q 59603307 IC50 = 110 nM T37848 CIDZ57 59603310 IC50 = 52 nM T37848 CJN23U 59603311 IC50 = 22 nM T37848 C6LZH4 59603314 IC50 = 60 nM T37848 CN8CA9 59603317 IC50 = 200 nM T37848 CM6T3L 59603319 IC50 = 26 nM T37848 C9BX3W 59603320 IC50 = 79 nM T37848 CXEH74 59603321 IC50 = 37 nM T37848 CKZ9Y2 59603322 IC50 = 23 nM T37848 CZ9X8Q 59603324 IC50 = 38 nM T37848 C2CT6F 59603325 IC50 = 140 nM T37848 CNVE86 59603326 IC50 = 55 nM T37848 CA57EU 59603328 IC50 = 92 nM T37848 CQ61DL 59603329 IC50 = 200 nM T37848 C15WPY 59603332 IC50 = 26 nM T37848 CB93QS 59603333 IC50 = 41 nM T37848 CX3MD2 59603334 IC50 = 44 nM T37848 CPR8Y3 59603336 IC50 = 39 nM T37848 CU2QL1 59603337 IC50 = 24 nM T37848 C8R0JT 59606002 IC50 > 10000 nM T37848 C9PL4C 59620419 IC50 = 560 nM T37848 C1W6VL 59620422 IC50 = 240 nM T37848 CT52DP 59620461 IC50 = 840 nM T37848 CP2UY3 59634686 IC50 > 27000 nM T37848 CPA0L2 59634709 IC50 > 27000 nM T37848 CPJ8R9 59635628 IC50 = 3500 nM T37848 CLSO80 59635752 IC50 = 10500 nM T37848 CS80HW 59648012 IC50 = 4900 nM T37848 C3RB0E 59648133 IC50 > 50000 nM T37848 CYKF93 59651916 IC50 > 30000 nM T37848 C5PDB3 59651957 IC50 > 30000 nM T37848 C4W8RH 59651989 IC50 > 30000 nM T37848 CV3I8D 59721232 IC50 = 500 nM T37848 CU1WE8 59721235 IC50 = 100 nM T37848 C6DZ9Q 59721239 IC50 = 130 nM T37848 CK4CL8 59721245 IC50 = 140 nM T37848 CT13LJ 59721254 IC50 = 120 nM T37848 CBEG02 59721267 IC50 = 190 nM T37848 CV6L5Y 59721273 IC50 = 140 nM T37848 CQ1DY2 59721278 IC50 = 150 nM T37848 CJ3Q8X 59721296 IC50 = 210 nM T37848 CS5U7D 59721308 IC50 = 210 nM T37848 C2E1VC 59721310 IC50 = 280 nM T37848 C9PFU4 59721343 IC50 = 130 nM T37848 CZ7B2I 59721348 IC50 = 130 nM T37848 COI87D 59721361 IC50 = 140 nM T37848 COG08J 59721362 IC50 = 120 nM T37848 CY01EP 59721363 IC50 = 150 nM T37848 CDV2Y4 59721364 IC50 = 80 nM T37848 CH35VM 59721369 IC50 < 100 nM T37848 C7SEC1 59721372 IC50 = 510 nM T37848 CT19BJ 59721374 IC50 = 710 nM T37848 CXU0N5 59721379 IC50 = 410 nM T37848 C06GAY 59721381 IC50 = 170 nM T37848 C2LQN0 59721382 IC50 = 140 nM T37848 CL5WT4 59721395 IC50 = 150 nM T37848 C8FB0T 59721398 IC50 = 140 nM T37848 C2M0TL 59721405 IC50 = 130 nM T37848 CK2UR9 59721409 IC50 = 110 nM T37848 C4I3JA 59721419 IC50 = 90 nM T37848 C7ECU2 59794447 IC50 > 40000 nM T37848 C63REN 59825673 IC50 = 190 nM T37848 C3UW1D 59825681 IC50 = 23000 nM T37848 C9LWV7 59825704 IC50 = 8400 nM T37848 CO34FC 59825742 IC50 = 170 nM T37848 C65BUA 59825756 IC50 = 12000 nM T37848 CI8C9G 59825774 IC50 = 1000 nM T37848 CZ8S5M 59825775 IC50 = 34000 nM T37848 C2W1TF 60001863 IC50 > 50000 nM T37848 CZE5J8 60026377 IC50 = 100 nM T37848 CJ34GW 60026481 IC50 = 2000 nM T37848 CJ7E6C 60026483 IC50 = 3000 nM T37848 C31PTC 60026641 IC50 = 100 nM T37848 CI36XS 60026787 IC50 = 200 nM T37848 C3JD8M 60026802 IC50 = 100 nM T37848 C3UQ8M 60026849 IC50 = 500 nM T37848 CM3Y0X 60026895 IC50 = 600 nM T37848 CE37AG 60097359 IC50 = 2000 nM T37848 CMF42W 60097605 IC50 = 480 nM T37848 C02BUA 60097693 IC50 = 10000 nM T37848 C9QRX3 60098131 IC50 = 1800 nM T37848 C5QS4J 60148513 IC50 = 3000 nM T37848 C4MV2N 60149678 IC50 > 30000 nM T37848 CTL97W 60151476 IC50 > 45000 nM T37848 C62SQG 60155628 IC50 > 20000 nM T37848 COS39T 60155629 IC50 > 10000 nM T37848 CE5A7B 60162406 IC50 > 22000 nM T37848 CWC26U 60165513 IC50 < 100 nM T37848 C67TFB 60165514 IC50 > 10000 nM T37848 CPL1G3 60165805 IC50 > 10000 nM T37848 C2D3HQ 60168069 IC50 > 30000 nM T37848 CI7U5V 60168601 IC50 = 3000 nM T37848 CLOU21 60169888 IC50 = 1000 nM T37848 CLES05 60170345 IC50 = 700 nM T37848 CBN9Y0 60170521 IC50 = 700 nM T37848 C2CKR1 60170522 IC50 = 1330 nM T37848 C2B0NS 60172115 IC50 = 3900 nM T37848 CIJ16Y 60196616 IC50 = 3800 nM T37848 C3S1RP 60197614 IC50 > 30000 nM T37848 CS4F2O 60197712 IC50 > 30000 nM T37848 C87HTO 60197713 IC50 > 30000 nM T37848 C5ES4W 60197714 IC50 = 16400 nM T37848 CF19XN 60197716 IC50 > 30000 nM T37848 COI61M 60197822 IC50 > 30000 nM T37848 CP1CK0 60197823 IC50 = 27400 nM T37848 C0JL3I 60197824 IC50 = 2000 nM T37848 CVOF90 60197825 IC50 = 8000 nM T37848 CBN3G4 60197937 IC50 > 30000 nM T37848 CS1WL6 60202315 IC50 = 1950 nM T37848 C7SGT6 60202316 IC50 = 14800 nM T37848 CT26JV 60202329 IC50 > 50000 nM T37848 CE18JH 60202715 IC50 = 285 nM T37848 CTO6J5 60203901 IC50 > 50000 nM T37848 CWA0B6 60204017 IC50 > 30000 nM T37848 C70EXD 60207864 IC50 = 1000 nM T37848 CW3H0V 60634975 IC50 > 25000 nM T37848 C4BZ2N 60637368 IC50 > 25000 nM T37848 CV13OQ 62705051 IC50 = 100 nM T37848 C9F4JW 62705832 IC50 < 2500 nM T37848 C04YCI 62706660 IC50 = 22 nM T37848 CKYT32 62706819 IC50 = 410 nM T37848 CXQR70 62706820 IC50 = 140 nM T37848 CH4U0K 62706821 IC50 = 42 nM T37848 C64RUV 62706976 IC50 = 2700 nM T37848 C24QGS 62707113 IC50 = 24 nM T37848 CX4N0I 62707515 IC50 = 90000 nM T37848 CJ5HI6 66547425 IC50 < 1000 nM T37848 CH76RD 66550504 IC50 > 25000 nM T37848 C2LBW7 66551925 IC50 > 50000 nM T37848 CLHX28 66553128 IC50 > 20000 nM T37848 C91JZL 66553214 IC50 = 40000 nM T37848 CNDH38 66557868 IC50 > 10000 nM T37848 CLRC36 66557875 IC50 > 30000 nM T37848 CUC7B3 66557964 IC50 > 30000 nM T37848 C1LB6D 66558197 IC50 = 1700 nM T37848 C7UKS4 66558379 IC50 = 5000 nM T37848 CCK6E5 66558639 IC50 = 510 nM T37848 C0G3LA 66559847 IC50 = 90000 nM T37848 C23NWU 66562843 IC50 = 9000 nM T37848 CE2S6P 66562938 IC50 = 8400 nM T37848 CK9FO4 66562947 IC50 = 1000 nM T37848 C1WXS5 66563037 IC50 = 2800 nM T37848 CG34JD 66563137 IC50 > 20000 nM T37848 C6LVU1 66563478 IC50 = 1000 nM T37848 C7FX5M 66563570 IC50 = 2000 nM T37848 C24BOR 66563571 IC50 = 1000 nM T37848 CQY3J2 66563572 IC50 = 3700 nM T37848 CY81CB 66575661 IC50 = 6000 nM T37848 CMXA10 66575743 IC50 > 50000 nM T37848 CBP6I7 66576773 IC50 > 50000 nM T37848 CZF76R 66608383 IC50 > 30000 nM T37848 CS72TK 66610926 IC50 > 10000 nM T37848 CVB4T1 66611375 IC50 > 10000 nM T37848 CUP41L 66613450 IC50 >= 30000 nM T37848 CFI5T8 66613669 IC50 = 7900 nM T37848 CCN98R 66649578 IC50 = 100 nM T37848 CHS2G5 66649612 IC50 = 3600 nM T37848 C75DVR 66649674 IC50 = 100 nM T37848 C2BGY7 66649788 IC50 = 1100 nM T37848 CY9TD4 66730677 IC50 > 10000 nM T37848 CJFS84 66731186 IC50 > 10000 nM T37848 CG1O8H 66734740 IC50 > 10000 nM T37848 C8CLK2 66735127 IC50 > 10000 nM T37848 CL5GH9 66735487 IC50 > 10000 nM T37848 CKN2U0 66764813 IC50 > 30000 nM T37848 CF15KL 66771109 IC50 > 50000 nM T37848 C51XCV 66781377 IC50 > 10000 nM T37848 CU6E0A 66818541 IC50 > 30000 nM T37848 CKD8I1 66818569 IC50 > 30000 nM T37848 C5LU1Z 66818766 IC50 > 30000 nM T37848 C5J4MR 66850717 IC50 > 10000 nM T37848 CC6JF4 66851197 IC50 = 7200 nM T37848 C40FKD 66898172 IC50 > 50000 nM T37848 C7TJ9X 66898814 IC50 > 50000 nM T37848 CX1P8I 67042254 IC50 > 25000 nM T37848 CFM6H7 67049587 IC50 > 100000 nM T37848 CH39DP 67053383 IC50 = 26000 nM T37848 C3LF8O 67053425 IC50 = 14000 nM T37848 C4NX6W 67070065 IC50 > 50000 nM T37848 CN8AS7 67072266 IC50 < 200000 nM T37848 CVT35R 67097557 IC50 = 1800 nM T37848 CSQ3J1 67098421 IC50 < 400 nM T37848 CJV8O4 67098558 IC50 = 1700 nM T37848 CE49GC 67098566 IC50 = 4500 nM T37848 COD28B 67098794 IC50 = 1600 nM T37848 C23QPJ 67098846 IC50 = 1600 nM T37848 C13OVI 67098869 IC50 = 7200 nM T37848 C9KQT3 67098926 IC50 = 1400 nM T37848 C52XBW 67098971 IC50 = 1200 nM T37848 CQ97ZW 67161103 IC50 = 25000 nM T37848 CNP52W 67163022 IC50 = 23000 nM T37848 CT9AH0 67178880 IC50 = 1400 nM T37848 CLU63M 67270136 IC50 = 100 nM T37848 CK16WC 67270717 IC50 = 100 nM T37848 C9AQ0T 67270792 IC50 = 160 nM T37848 CVL03S 67270914 IC50 = 400 nM T37848 C8EFI1 67270974 IC50 = 100 nM T37848 CY76UR 67305743 IC50 = 20000 nM T37848 C3UKG8 67312397 IC50 > 10000 nM T37848 CM6TZ3 67312506 IC50 = 18000 nM T37848 CKMV48 67345882 IC50 > 10000 nM T37848 C50IMJ 67387021 IC50 > 20000 nM T37848 C36MVU 67389741 IC50 = 11300 nM T37848 C4R8OG 67401728 IC50 > 30000 nM T37848 CX8JP5 67402849 IC50 > 40000 nM T37848 CPV39L 67406727 IC50 > 30000 nM T37848 C4S3FE 67450880 IC50 = 67000 nM T37848 C8L5HO 67453320 IC50 > 100000 nM T37848 C37YHJ 67496729 IC50 > 30000 nM T37848 C9AIK4 67522993 IC50 = 170 nM T37848 CNB15W 67607112 IC50 = 1100 nM T37848 C1UE3F 67928759 IC50 > 10000 nM T37848 CE94JQ 67953283 IC50 > 50000 nM T37848 CT43SM 67953330 IC50 > 50000 nM T37848 CPTA39 67953837 IC50 > 50000 nM T37848 CD3HT9 67960134 IC50 > 25000 nM T37848 CAF36T 67972044 IC50 = 1000 nM T37848 C5K7QG 67974411 IC50 >= 30000 nM T37848 CW7Y0S 68000593 IC50 > 27000 nM T37848 C4HEC3 68001087 IC50 > 27000 nM T37848 CO75NL 68011817 IC50 > 10000 nM T37848 CBOF40 68046989 IC50 > 50000 nM T37848 CGW5L9 68075088 IC50 > 30000 nM T37848 CN3KZ8 68161075 IC50 = 2000 nM T37848 CJ6N4O 68166092 IC50 = 120 nM T37848 C8JVH7 68166270 IC50 = 300 nM T37848 C32TVX 68230798 IC50 = 1000 nM T37848 C5YCB6 68234668 IC50 > 40000 nM T37848 CR17ZU 68234693 IC50 > 40000 nM T37848 CZCP37 68234870 IC50 > 100000 nM T37848 C9J8GY 68234878 IC50 > 40000 nM T37848 CN6KL0 68235029 IC50 = 11540 nM T37848 C1KAG4 68235232 IC50 > 40000 nM T37848 C7TR4I 68276577 IC50 = 5700 nM T37848 CK5V3O 68277611 IC50 > 10000 nM T37848 C17JAZ 68284084 IC50 > 30000 nM T37848 CCT07V 68290289 IC50 > 20000 nM T37848 C4LKB3 68291752 IC50 > 20000 nM T37848 CMG58Q 68295585 IC50 > 15000 nM T37848 CPA95O 68380152 IC50 > 30000 nM T37848 C95VPL 68380260 IC50 > 30000 nM T37848 CPW29C 68411962 IC50 = 34 nM T37848 C61SJG 68412618 IC50 = 90 nM T37848 C30WPU 68417067 IC50 = 250 nM T37848 CAB4M3 68447092 IC50 <= 200 nM T37848 C56CFA 68448803 IC50 = 2500 nM T37848 CVM9Q1 68503758 IC50 > 50000 nM T37848 CLS10P 68513301 IC50 = 6400 nM T37848 C5JYB8 68515257 IC50 > 20000 nM T37848 C69OHY 68560854 IC50 = 35000 nM T37848 CCD89X 68563058 IC50 = 80000 nM T37848 C48EIQ 68568011 IC50 > 100000 nM T37848 CH3Z7F 68658979 IC50 > 50000 nM T37848 CL6N2D 68775231 IC50 > 50000 nM T37848 C89CQS 68779277 IC50 > 10000 nM T37848 CNI8V4 68785998 IC50 = 480 nM T37848 CV4NO2 69080188 IC50 = 8700 nM T37848 CNJ7K2 69081619 IC50 = 1400 nM T37848 C4IW9J 69081640 IC50 = 6600 nM T37848 CJI32G 69081964 IC50 > 30000 nM T37848 C3RDA0 69082236 IC50 = 10000 nM T37848 COE39Z 69082854 IC50 = 25000 nM T37848 C6PR7O 69083435 IC50 = 5200 nM T37848 C97BGW 69093249 IC50 = 102000 nM T37848 CZC4E1 69093450 IC50 = 23000 nM T37848 C02UFD 69224054 IC50 > 17000 nM T37848 C7SQT4 69224555 IC50 = 20000 nM T37848 C7Z9LF 69224988 IC50 > 17000 nM T37848 C7ZX9P 69281312 IC50 >= 195000 nM T37848 C7PY1Q 69281314 IC50 = 14000 nM T37848 COJ4Q1 69315206 IC50 = 37000 nM T37848 CJ5Z7T 69316129 IC50 = 4000 nM T37848 CA49UK 69520512 IC50 = 13000 nM T37848 CNQ8T5 69571559 IC50 = 600 nM T37848 C67CPF 69576646 IC50 = 1000 nM T37848 C5VJG4 69643233 IC50 > 30000 nM T37848 CRM37W 69936689 IC50 < 100 nM T37848 CY73XK 69936726 IC50 = 4300 nM T37848 C7YIU0 69936777 IC50 = 6200 nM T37848 CHD80I 69937162 IC50 > 50000 nM T37848 CAR2N8 69937236 IC50 > 50000 nM T37848 CN7X0U 69937257 IC50 > 50000 nM T37848 CC8QU9 70227534 IC50 = 100 nM T37848 C06WFN 70276830 IC50 > 31622.78 nM T37848 CDQ85E 70276990 IC50 = 630.96 nM T37848 CS47OP 70496411 IC50 = 4600 nM T37848 CK5H1Y 70497007 IC50 > 10000 nM T37848 C6NSG3 70497750 IC50 > 10000 nM T37848 CWP52K 70497865 IC50 > 10000 nM T37848 C7VJ6A 70647728 IC50 > 40000 nM T37848 CFH68K 70664065 IC50 = 2400 nM T37848 CAR46Z 70675172 IC50 > 25000 nM T37848 C97WSO 70678458 IC50 > 30000 nM T37848 CC6T5K 70679283 IC50 > 30000 nM T37848 C0I7PG 70681152 IC50 > 33000 nM T37848 C7GJW9 70681170 IC50 = 4700 nM T37848 CAO1N7 70681171 IC50 = 1900 nM T37848 CC20VE 70681172 IC50 = 1900 nM T37848 C8H4JX 70681173 IC50 = 3900 nM T37848 C6NYK2 70681174 IC50 = 1700 nM T37848 C7W3JA 70681326 IC50 > 5000 nM T37848 CNA09E 70682193 IC50 = 30 nM T37848 C9S1RD 70682194 IC50 = 1300 nM T37848 C8XC1S 70682487 IC50 = 14200 nM T37848 CI8EQ5 70682492 IC50 = 1000 nM T37848 CPF92N 70682528 IC50 = 5600 nM T37848 C37CFL 70682529 IC50 = 7800 nM T37848 C8KBJ0 70683271 IC50 = 6100 nM T37848 CU5C2B 70684211 IC50 = 180 nM T37848 CMHV13 70684212 IC50 = 27 nM T37848 C1H8IU 70684268 IC50 = 130 nM T37848 CT94WJ 70684556 IC50 > 30000 nM T37848 CU1I5S 70684569 IC50 = 1000 nM T37848 CM96VS 70684570 IC50 = 1000 nM T37848 CZHB48 70684601 IC50 = 2900 nM T37848 C5P0CI 70684602 IC50 = 7700 nM T37848 C86ETQ 70684603 IC50 = 7000 nM T37848 CCM9Z5 70684604 IC50 > 20000 nM T37848 C4FH7S 70684606 IC50 > 20000 nM T37848 CHFM92 70685176 IC50 > 50000 nM T37848 CG6BY1 70685177 IC50 > 30000 nM T37848 CWIC42 70685308 IC50 > 10000 nM T37848 CU50BK 70685377 IC50 = 1500 nM T37848 C3MB6V 70685378 IC50 = 1800 nM T37848 C60SBP 70685515 IC50 > 9000 nM T37848 C3UO2F 70686000 IC50 = 100000 nM T37848 C9BQS5 70686347 IC50 = 200 nM T37848 CXMN06 70686415 IC50 = 140 nM T37848 CRA4G1 70686722 IC50 = 1000 nM T37848 C9V6ML 70687502 IC50 = 36000 nM T37848 C4VU7J 70688210 IC50 > 50000 nM T37848 CVFM91 70688283 IC50 > 200000 nM T37848 CHX94N 70688456 IC50 = 84 nM T37848 C6EKP1 70688461 IC50 = 97 nM T37848 C3B9AV 70688462 IC50 = 30 nM T37848 C54FUX 70688463 IC50 = 69 nM T37848 C4L2QN 70688512 IC50 = 53 nM T37848 CTKA58 70688513 IC50 = 38 nM T37848 CL4I8H 70688552 IC50 > 40000 nM T37848 CZC4Y2 70688845 IC50 = 10000 nM T37848 CE1GI4 70688847 IC50 = 5700 nM T37848 C18OFS 70688848 IC50 > 20000 nM T37848 CIF26X 70689554 IC50 = 17000 nM T37848 C4GXP2 70690453 IC50 > 30000 nM T37848 CN6TB1 70690521 IC50 = 31 nM T37848 C0YA3Z 70690615 IC50 = 2400 nM T37848 CFQ7Z0 70690616 IC50 = 100 nM T37848 C4BG7D 70690617 IC50 = 7300 nM T37848 CQ0SN9 70691313 IC50 = 4015 nM T37848 CH34MZ 70691697 IC50 = 2000 nM T37848 CXD3F9 70691699 IC50 = 3700 nM T37848 C0XRC9 70691981 IC50 > 8600 nM T37848 C7I2LV 70692667 IC50 = 30 nM T37848 CE46OL 70692716 IC50 = 33 nM T37848 CRDT90 70692759 IC50 = 30 nM T37848 C3DV6C 70693036 IC50 = 1000 nM T37848 CJ0P9G 70693067 IC50 = 20000 nM T37848 C8IOC9 70693068 IC50 = 5000 nM T37848 CF5YQ9 70693069 IC50 = 5900 nM T37848 CI4KP9 70693070 IC50 > 20000 nM T37848 CG4S9N 70693071 IC50 = 5100 nM T37848 C8G4AV 70694560 IC50 = 3100 nM T37848 CVH1E7 70694802 IC50 = 84 nM T37848 C1P7ZJ 70694804 IC50 < 1000 nM T37848 CC6GZ9 70695067 IC50 > 20000 nM T37848 CS1MU4 70695116 IC50 > 20000 nM T37848 C6K9BL 70695117 IC50 = 11000 nM T37848 C1YZ6K 70695118 IC50 = 6600 nM T37848 C53RQN 70695119 IC50 = 3800 nM T37848 CXJ5V2 70695120 IC50 = 2600 nM T37848 CCR12A 70695121 IC50 > 20000 nM T37848 CVU08A 70695812 IC50 > 25000 nM T37848 C37YJI 70695889 IC50 = 3100 nM T37848 C8Z2LD 70696754 IC50 = 37 nM T37848 C8QP2E 70696805 IC50 = 230 nM T37848 C6WM8C 70696806 IC50 = 120 nM T37848 CK42BQ 70696845 IC50 = 16000 nM T37848 C62EGB 70696847 IC50 > 40000 nM T37848 CV38GW 70697123 IC50 = 1000 nM T37848 CSX71G 70697153 IC50 = 14000 nM T37848 C4JY5R 70697154 IC50 = 5200 nM T37848 CT78JN 70697155 IC50 = 8700 nM T37848 C34WHG 70697225 IC50 = 3981.07 nM T37848 CBDL19 70792359 IC50 > 100000 nM T37848 C7DO1N 70817239 IC50 > 20000 nM T37848 C6L7FH 70817382 IC50 = 8000 nM T37848 C2PJ1D 70865101 IC50 > 30000 nM T37848 CUCQ24 70874317 IC50 = 2600 nM T37848 C8LCK6 70874412 IC50 = 10 nM T37848 C1H7VK 70874453 IC50 = 2000 nM T37848 CJF91M 70874544 IC50 = 1200 nM T37848 C9EWB8 70874603 IC50 = 10900 nM T37848 C82PUD 70874605 IC50 = 130 nM T37848 C8Q4LJ 70874786 IC50 = 60 nM T37848 CF1G3K 70874916 IC50 = 3300 nM T37848 C30AJI 70914208 IC50 = 1100 nM T37848 C71AZM 70914219 IC50 = 3800 nM T37848 C2TC8W 70914230 IC50 = 3100 nM T37848 C8V5NF 70914234 IC50 = 5600 nM T37848 CP8HI7 70914358 IC50 = 8600 nM T37848 CXW7U0 70977933 IC50 > 10000 nM T37848 C1VMF2 70977969 IC50 > 50000 nM T37848 CA6GI0 70993878 IC50 = 340 nM T37848 C1XHA8 71116039 IC50 = 40000 nM T37848 CQV38O 71143628 IC50 = 74000 nM T37848 C5BF7P 71143790 IC50 = 136000 nM T37848 C2HGI7 71153408 IC50 > 10000 nM T37848 C62ULC 71225056 IC50 > 100000 nM T37848 C7Y2LB 71230234 IC50 > 10000 nM T37848 C5RE4T 71244643 IC50 > 10000 nM T37848 C9AT8D 71263621 IC50 = 4200 nM T37848 C6BE5X 71271461 IC50 > 50000 nM T37848 C47QTF 71279423 IC50 > 50000 nM T37848 CH4T8Z 71279444 IC50 > 50000 nM T37848 C4E1RT 71279494 IC50 > 50000 nM T37848 CZR37K 71279507 IC50 > 50000 nM T37848 CU4P3X 71279543 IC50 > 50000 nM T37848 C5L8SW 71279563 IC50 > 50000 nM T37848 CQ7L0A 71279608 IC50 > 19000 nM T37848 CXZG59 71280008 IC50 > 50000 nM T37848 C5TXH9 71280067 IC50 > 50000 nM T37848 CW0FK6 71280128 IC50 > 50000 nM T37848 CEO08K 71280143 IC50 > 50000 nM T37848 C5CTH0 71280416 IC50 > 50000 nM T37848 CHY7N4 71280456 IC50 > 19000 nM T37848 C3LOB1 71285746 IC50 > 50000 nM T37848 C7PLS6 71285927 IC50 > 50000 nM T37848 C68LPJ 71288456 IC50 > 7000 nM T37848 C7MPQ3 71288593 IC50 = 37000 nM T37848 CW1UG2 71288611 IC50 = 1600 nM T37848 CL3E4J 71288616 IC50 = 25000 nM T37848 CP89XV 71288634 IC50 = 1900 nM T37848 CM8L7K 71288636 IC50 = 7700 nM T37848 C5ARM6 71288638 IC50 = 14000 nM T37848 C29CFW 71288697 IC50 = 2700 nM T37848 CD7R9M 71288713 IC50 = 7800 nM T37848 CPQ95B 71288715 IC50 = 15000 nM T37848 CNC5Z3 71288739 IC50 = 17000 nM T37848 C18JBK 71288740 IC50 = 3200 nM T37848 C0QOF3 71288752 IC50 = 54000 nM T37848 CW31HT 71288754 IC50 = 2700 nM T37848 CP1H9R 71291709 IC50 = 770 nM T37848 CAO07V 71293843 IC50 = 2070 nM T37848 CWN2M1 71300316 IC50 > 30000 nM T37848 C03KNO 71300317 IC50 > 30000 nM T37848 CWY4S0 71304814 IC50 > 50000 nM T37848 CS9OV5 71315139 Ki = 120 nM T37848 CR37DA 71419478 IC50 = 12589.25 nM T37848 C5SML3 71449452 IC50 = 15848.93 nM T37848 CL6BC1 71449606 IC50 = 1600 nM T37848 CR46HB 71449876 IC50 = 15 nM T37848 CB6F1U 71450284 IC50 = 6300 nM T37848 C1C6UV 71450309 IC50 = 30 nM T37848 CCL8I2 71451192 IC50 = 25000000 nM T37848 CCR9W0 71451887 IC50 = 2800 nM T37848 CY3ZK1 71452107 IC50 = 10700 nM T37848 C9QKH0 71452111 IC50 = 5800 nM T37848 COQ0P1 71453071 IC50 = 12589.25 nM T37848 C6VY5W 71453938 IC50 = 7000 nM T37848 CXEQ42 71453953 IC50 = 100 nM T37848 CSL01M 71454248 IC50 = 5011.87 nM T37848 C47GYB 71454279 IC50 > 10000 nM T37848 CJM13D 71454747 IC50 = 25000000 nM T37848 CJ6T7O 71455231 IC50 = 15 nM T37848 C0YD9K 71455398 IC50 = 2000 nM T37848 CR9VU6 71455427 IC50 = 6000 nM T37848 C5KYQ3 71455673 IC50 = 4300 nM T37848 C84KML 71455676 IC50 = 1500 nM T37848 C4O2GZ 71457203 IC50 = 1900 nM T37848 C7MNB5 71457264 IC50 = 6460 nM T37848 CH6Q3P 71457466 IC50 = 100 nM T37848 CCFZ37 71457467 IC50 = 30 nM T37848 C14SIK 71459316 IC50 = 10900 nM T37848 C8W1GO 71459317 IC50 = 6700 nM T37848 C5BZ6H 71459318 IC50 = 10600 nM T37848 C3WZ8U 71459328 IC50 = 7900 nM T37848 CN8I4U 71459342 IC50 = 50 nM T37848 C0NJ6Y 71460877 IC50 > 30000 nM T37848 CSZE81 71461095 IC50 = 9200 nM T37848 CS0XO4 71461098 IC50 = 9400 nM T37848 CH72YK 71461109 IC50 = 30 nM T37848 CBMS65 71461110 IC50 = 30 nM T37848 CW1X7I 71461437 IC50 = 1100 nM T37848 C64WKU 71462837 IC50 = 8300 nM T37848 CD81EJ 71463058 IC50 = 200 nM T37848 C0GBL7 71466345 IC50 > 20000 nM T37848 CT08NF 71475689 IC50 = 72000 nM T37848 CC3N4O 71492530 IC50 = 1300 nM T37848 C3G9YK 71494647 IC50 = 10000 nM T37848 CFA9V1 71494937 IC50 > 33000 nM T37848 CCV93P 71506845 IC50 = 28600 nM T37848 C8U0TA 71510812 IC50 > 25000 nM T37848 C9DIK2 71512060 IC50 > 10000 nM T37848 CF05BU 71513157 IC50 > 10000 nM T37848 CS1ZX0 71513822 IC50 > 10000 nM T37848 C0VLE3 71516457 IC50 > 20000 nM T37848 C2LVY0 71516458 IC50 > 20000 nM T37848 CA07TC 71517197 IC50 > 10000 nM T37848 C7Q8ST 71522361 IC50 > 50000 nM T37848 C9JQ3C 71525043 IC50 = 360 nM T37848 CNFJ29 71525169 IC50 = 10 nM T37848 CD26MN 71525170 IC50 = 1 nM T37848 C06DJE 71525218 IC50 = 30 nM T37848 C1OF9Y 71525219 IC50 = 360 nM T37848 C83BHF 71525220 IC50 = 2600 nM T37848 C9KRS5 71525221 IC50 = 10000 nM T37848 C5VG9H 71525222 IC50 = 2300 nM T37848 CJE5P1 71525223 IC50 = 3000 nM T37848 CNI98B 71525653 IC50 > 20000 nM T37848 C3CT1R 71530223 IC50 = 7500 nM T37848 CN8CM1 71533722 IC50 = 50000 nM T37848 CPZ5S8 71535400 IC50 = 3500 nM T37848 CCRS95 71535683 IC50 > 50000 nM T37848 CRU94Y 71536970 IC50 = 14500 nM T37848 CW8U2R 71537836 IC50 = 18600 nM T37848 C1SM3T 71539661 Ki = 1160 nM T37848 C67ZSQ 71540073 IC50 > 30000 nM T37848 C3RQP5 71542927 IC50 > 10000 nM T37848 C1GUX2 71542931 IC50 > 10000 nM T37848 C0IK7U 71544354 IC50 > 12.5 nM T37848 C9N7YA 71544706 IC50 = 8800 nM T37848 C92NEY 71544707 IC50 > 20000 nM T37848 C83YJF 71544946 IC50 > 50000 nM T37848 C4N3OC 71545856 IC50 = 5500 nM T37848 CCN01X 71547862 IC50 > 10000 nM T37848 CKB12X 71549359 IC50 = 30000 nM T37848 C4LZM6 71549637 IC50 = 11000 nM T37848 C6JOB5 71549767 IC50 = 55000 nM T37848 CV47CJ 71549769 IC50 = 80000 nM T37848 C5IV9D 71549913 IC50 = 45000 nM T37848 CSHT69 71550657 IC50 > 19000 nM T37848 CHO7D1 71555244 IC50 = 3900 nM T37848 CM04ZX 71555465 IC50 = 380 nM T37848 C5HK2E 71555534 IC50 = 780 nM T37848 C9P5KT 71556166 IC50 > 50000 nM T37848 C8JOU5 71556223 IC50 > 50000 nM T37848 C25XGY 71556353 IC50 > 50000 nM T37848 CP0J5L 71556425 IC50 > 50000 nM T37848 CB5QR3 71556493 IC50 = 16000 nM T37848 CIXL34 71556883 IC50 > 50000 nM T37848 CZ3A7E 71556887 IC50 > 50000 nM T37848 CY59CA 71557630 IC50 = 150 nM T37848 CTI52S 71557789 IC50 = 140 nM T37848 CMKH30 71558122 IC50 > 10000 nM T37848 CS8M1O 71558621 IC50 > 10000 nM T37848 CJXK67 71559365 IC50 = 77 nM T37848 C30ZKJ 71561420 IC50 > 10000 nM T37848 CS2VA3 71569375 IC50 = 1600 nM T37848 C9WNA4 71569533 IC50 = 7300 nM T37848 C4MO6G 71571541 IC50 = 870 nM T37848 C2L8XG 71572646 IC50 > 20000 nM T37848 CLR92N 71579539 IC50 = 6900 nM T37848 C84GAB 71580631 IC50 = 5100 nM T37848 C4S1TN 71580827 IC50 = 1500 nM T37848 C6CHY1 71580912 IC50 = 6500 nM T37848 CUJT21 71582799 IC50 > 10000 nM T37848 CWD2Z5 71585566 IC50 > 10000 nM T37848 CCE7T2 71585568 IC50 > 10000 nM T37848 C6L4DN 71602354 IC50 = 64000 nM T37848 C0WAH3 71602807 IC50 = 26000 nM T37848 CT9DI2 71603188 IC50 > 100000 nM T37848 C9MIF7 71603190 IC50 = 7900 nM T37848 CD87XO 71603193 IC50 > 100000 nM T37848 C9J0EH 71603917 IC50 > 50000 nM T37848 C13FGZ 71604895 IC50 > 10000 nM T37848 CNY35F 71604897 IC50 = 5000 nM T37848 CN08ZO 71605054 IC50 = 7300 nM T37848 C4D8XS 71621494 IC50 > 200000 nM T37848 CD7OB1 71621495 IC50 > 200000 nM T37848 CBQT67 71621649 IC50 > 200000 nM T37848 CD3FK8 71621650 IC50 = 198000 nM T37848 C3Y4VO 71621800 IC50 > 200000 nM T37848 CCP1M5 71621802 IC50 > 200000 nM T37848 CKPV51 71621803 IC50 > 200000 nM T37848 CLA5F0 71622218 IC50 > 200000 nM T37848 CTY84A 71622350 IC50 > 200000 nM T37848 C8SGK6 71624246 IC50 = 9950 nM T37848 C2WJX0 71626755 IC50 > 50000 nM T37848 C26TXG 71626895 IC50 > 50000 nM T37848 C4DHC9 71626896 IC50 > 50000 nM T37848 CX0VE7 71626971 IC50 > 50000 nM T37848 CDL35U 71655748 IC50 > 5000 nM T37848 CAN6X5 71656574 IC50 = 43000 nM T37848 C61RYH 71659356 IC50 > 30000 nM T37848 CVDB58 71659357 IC50 > 30000 nM T37848 C28EIT 71659358 IC50 > 30000 nM T37848 C8DF4B 71659489 IC50 > 30000 nM T37848 C7Y0RM 71659490 IC50 > 30000 nM T37848 CKR47S 71659491 IC50 > 30000 nM T37848 CAQ2V1 71659492 IC50 > 30000 nM T37848 CJX32Y 71659493 IC50 > 30000 nM T37848 C05JLG 71659494 IC50 > 30000 nM T37848 COS6Q5 71659610 IC50 > 30000 nM T37848 CNVI07 71659611 IC50 > 30000 nM T37848 CUF06Z 71659612 IC50 > 30000 nM T37848 CT9KZ0 71659613 IC50 > 30000 nM T37848 CZFU74 71659614 IC50 > 30000 nM T37848 CC3L1Y 71659615 IC50 > 30000 nM T37848 CF1HA9 71659751 IC50 = 24000 nM T37848 CF8DV2 71659752 IC50 > 30000 nM T37848 CMA4N0 71659753 IC50 > 30000 nM T37848 CFBA41 71659754 IC50 > 30000 nM T37848 CR58TZ 71659755 IC50 > 30000 nM T37848 CVE91N 71659756 IC50 > 30000 nM T37848 CH4VF0 71659894 IC50 > 30000 nM T37848 C53AOG 71659895 IC50 > 30000 nM T37848 C9WC2J 71659896 IC50 > 30000 nM T37848 CTBX46 71659897 IC50 = 7500 nM T37848 CW0Y5N 71659898 IC50 > 30000 nM T37848 CZD71P 71680760 IC50 = 7000 nM T37848 CZ1H8S 71681176 IC50 > 27000 nM T37848 C2RGP3 71681329 IC50 = 7600 nM T37848 CI5E8F 71681330 IC50 = 5400 nM T37848 CCXO28 71681727 IC50 = 1800 nM T37848 C23QGT 71681728 IC50 = 710 nM T37848 CU20IN 71681888 IC50 > 30000 nM T37848 CR29TS 71681889 IC50 = 980 nM T37848 CC7MT2 71681890 IC50 = 15000 nM T37848 CF7R0Y 71682057 IC50 > 30000 nM T37848 C4LO5V 71682058 IC50 > 30000 nM T37848 CM78WZ 71682209 IC50 > 30000 nM T37848 CMG8N0 71682210 IC50 = 17000 nM T37848 CRN3A6 71682211 IC50 > 30000 nM T37848 CX48CN 71682212 IC50 = 7700 nM T37848 C0EMZ1 71682213 IC50 = 17000 nM T37848 CQ53SW 71682214 IC50 > 30000 nM T37848 CWG8M3 71682651 IC50 > 10000 nM T37848 CY8VM4 71695585 IC50 > 10000 nM T37848 C8LE5D 71695973 IC50 > 10000 nM T37848 C9I3GO 71714121 IC50 = 18000 nM T37848 CC4A3K 71716821 IC50 = 616 nM T37848 CUG2V3 71716866 IC50 = 556 nM T37848 CIZ40M 71716873 IC50 > 30000 nM T37848 C56LUJ 71716957 IC50 > 50000 nM T37848 C4XYN9 71717494 IC50 > 30000 nM T37848 C5K9JV 71717638 IC50 = 5000 nM T37848 C89GSF 71718127 IC50 = 15124 nM T37848 CWB3V1 71718136 IC50 = 6800 nM T37848 C7TM8H 71718630 IC50 > 30000 nM T37848 CW38FM 71718726 IC50 < 30 nM T37848 CS8CZ7 71718968 IC50 > 50000 nM T37848 CY6D2J 71719903 IC50 = 26588 nM T37848 CL0O5N 71719912 IC50 = 400 nM T37848 CYQH30 71719914 IC50 = 11068 nM T37848 C86MQI 71720046 IC50 > 10000 nM T37848 C1FYA8 71720426 IC50 > 20000 nM T37848 CMDI34 71720470 IC50 = 910 nM T37848 C7B8UH 71720543 IC50 = 205 nM T37848 CA9Y3R 71720882 IC50 = 15000 nM T37848 C5UBH0 71720883 IC50 > 20000 nM T37848 CQEH46 71720911 IC50 = 90 nM T37848 C30NBJ 71722055 IC50 > 10000 nM T37848 CIN10C 71727133 IC50 > 10000 nM T37848 COI5S0 71727368 IC50 = 340 nM T37848 CB53IQ 71727461 IC50 > 10000 nM T37848 CLE15B 71727801 IC50 > 10000 nM T37848 C6USH8 71727930 IC50 > 10000 nM T37848 C1W4DX 71727932 IC50 > 10000 nM T37848 CJZR51 71728054 IC50 > 10000 nM T37848 C5TS9Y 71731356 IC50 = 97900 nM T37848 CD9F5X 71731476 IC50 = 79360 nM T37848 C3IO9H 71731477 IC50 = 91930 nM T37848 CVAD62 71731478 IC50 = 58280 nM T37848 C1ON0X 71731479 IC50 = 46240 nM T37848 CZYQ05 71731604 IC50 = 42190 nM T37848 C40YRO 71731605 IC50 = 54650 nM T37848 CQ21ZD 71733911 IC50 > 50000 nM T37848 C56MYK 71739468 IC50 > 30000 nM T37848 CH45ZR 71744719 IC50 > 20000 nM T37848 C60BIX 71763463 IC50 > 10000 nM T37848 C5CDM4 71766212 IC50 > 20000 nM T37848 C6P9HZ 71766360 IC50 > 20000 nM T37848 CJHI28 71770158 IC50 = 6 nM T37848 C9LU5Q 71770282 IC50 = 1450 nM T37848 CTSK68 71811225 IC50 = 6500 nM T37848 CVL54T 71811261 IC50 = 100 nM T37848 CH8M5Y 71811363 IC50 > 50000 nM T37848 C1WT8V 71811365 IC50 > 50000 nM T37848 COVS02 71812189 IC50 > 30000 nM T37848 C5JV1P 71812623 EC50 > 100000 nM T37848 CJH9K3 71814859 IC50 > 10000 nM T37848 CD28XR 71816087 IC50 > 10000 nM T37848 CC4SU1 71817351 IC50 > 10000 nM T37848 CY04LE 71817500 IC50 > 10000 nM T37848 CX0WV5 71817943 IC50 = 1759 nM T37848 CN1LU6 71817944 IC50 > 10000 nM T37848 CGV4U3 71817945 IC50 = 1262 nM T37848 CJ4L5G 71818086 IC50 = 1009 nM T37848 COXA51 71818087 IC50 > 10000 nM T37848 CP1A3M 71818088 IC50 > 10000 nM T37848 CPJ42T 71818089 IC50 = 3581 nM T37848 CAP03I 71818090 IC50 > 10000 nM T37848 CO23PK 71818091 IC50 = 4196 nM T37848 CL4X6A 71818092 IC50 = 6720 nM T37848 CL8GK5 71818093 IC50 = 5046 nM T37848 C4ZVG0 71818094 IC50 > 10000 nM T37848 CH2GR0 71818232 IC50 = 1739 nM T37848 C0VGQ9 71818233 IC50 > 10000 nM T37848 C5QRF2 71818234 IC50 = 2145 nM T37848 C2K0CS 71819719 IC50 = 10200 nM T37848 C6EC3O 72163432 IC50 = 6200 nM T37848 CNF81W 72163837 IC50 > 30000 nM T37848 CB2NP7 72165228 IC50 > 20000 nM T37848 C2OV4Z 72189207 IC50 > 10000 nM T37848 CW4E9O 72189514 IC50 > 10000 nM T37848 CAVB46 72189515 IC50 > 10000 nM T37848 C4KUM3 72189516 IC50 > 10000 nM T37848 CR5Y6U 72189517 IC50 > 10000 nM T37848 C46FSX 72189518 IC50 > 10000 nM T37848 CBW0G9 72189519 IC50 > 10000 nM T37848 CC0DB5 72189807 IC50 > 10000 nM T37848 CUQ69N 72189808 IC50 > 10000 nM T37848 C1V7PU 72189809 IC50 > 10000 nM T37848 CC1SR3 72189810 IC50 > 10000 nM T37848 C9NCE7 72189811 IC50 > 10000 nM T37848 C2ZF9X 72190130 IC50 > 10000 nM T37848 CXH2S6 72190131 IC50 > 10000 nM T37848 C12KEZ 72190132 IC50 > 10000 nM T37848 CW64OR 72190133 IC50 > 10000 nM T37848 C9UV7C 72190738 IC50 > 10000 nM T37848 CZ60LS 72191037 IC50 = 300 nM T37848 C14GNR 72191038 IC50 = 300 nM T37848 C20HKS 72191344 IC50 = 700 nM T37848 CYEI57 72191660 IC50 = 1000 nM T37848 C36QKA 72191661 IC50 = 2400 nM T37848 C1Y8VS 72191976 IC50 = 900 nM T37848 CO28LK 72191977 IC50 = 4700 nM T37848 C5ZGJ6 72191978 IC50 = 1600 nM T37848 CWT7K2 72205601 IC50 = 80 nM T37848 CJHR52 72374726 IC50 = 1300 nM T37848 C9Z2XS 72374727 IC50 = 700 nM T37848 C1R7NT 72374728 IC50 = 1700 nM T37848 CTKQ98 72375000 IC50 > 30000 nM T37848 CL15CY 72375001 IC50 > 30000 nM T37848 CM92XP 72375119 IC50 > 30000 nM T37848 CE46KA 72375120 IC50 > 30000 nM T37848 CHVL93 72375121 IC50 > 30000 nM T37848 C1T4OK 72375745 IC50 = 2200 nM T37848 CSGV46 72376194 IC50 = 1900 nM T37848 CDEN65 72543942 IC50 > 27000 nM T37848 CR9F6I 72543943 IC50 > 27000 nM T37848 CK7DE4 72545105 IC50 > 20000 nM T37848 CA7Y1S 72547022 IC50 = 13000 nM T37848 CW24CT 72547023 IC50 = 27000 nM T37848 C2NCW7 72547024 IC50 > 27000 nM T37848 C7W9JZ 72547025 IC50 = 15300 nM T37848 C1I6VN 72547026 IC50 = 100 nM T37848 CU80HY 72547065 IC50 > 30000 nM T37848 CE3X8Y 72547066 IC50 > 30000 nM T37848 CCVG84 72547070 IC50 > 30000 nM T37848 C0Y6IK 72547282 IC50 > 27000 nM T37848 CK50CR 72547283 IC50 = 600 nM T37848 CZI51W 72547284 IC50 = 16200 nM T37848 C3PTC5 72547285 IC50 = 3500 nM T37848 CY5DQ1 72547286 IC50 = 4700 nM T37848 C5XCD4 72547287 IC50 > 27000 nM T37848 CX70JT 72547320 IC50 > 30000 nM T37848 CPSB14 72547529 IC50 = 2200 nM T37848 CY91WF 72547530 IC50 = 4500 nM T37848 C48CJQ 72547531 IC50 = 12200 nM T37848 CGTC61 72547532 IC50 > 27000 nM T37848 C81YEF 72547533 IC50 > 27000 nM T37848 C2Q6YJ 72670421 IC50 > 50000 nM T37848 C4G2UR 72695027 IC50 > 10000 nM T37848 CDFO42 72695136 IC50 > 10000 nM T37848 CK7F6U 72700776 IC50 > 10000 nM T37848 CM75FY 72703989 IC50 > 25000 nM T37848 CPQ34Z 72703991 IC50 > 25000 nM T37848 CBE48L 72707143 IC50 > 10000 nM T37848 C7ARW4 72707537 IC50 = 14080 nM T37848 CCW09H 72710598 IC50 = 1500 nM T37848 C9OQ2I 72710839 IC50 = 3000 nM T37848 CV5FZ2 72711021 IC50 = 15000 nM T37848 CB41XI 72711023 IC50 = 3300 nM T37848 C8AJW5 72711027 IC50 = 1500 nM T37848 CE5TM6 72711029 IC50 = 1100 nM T37848 CZ0RU4 72711249 IC50 = 1200 nM T37848 C3SGZ4 72711251 IC50 = 1500 nM T37848 CA6U8Q 72711253 IC50 = 1200 nM T37848 C7I9ZM 72711255 IC50 = 860 nM T37848 CJF4B2 72711479 IC50 = 1400 nM T37848 CNA70E 72711481 IC50 = 2000 nM T37848 CB09LR 72711483 IC50 = 1800 nM T37848 C2LCM8 72711720 IC50 = 1200 nM T37848 C95UWO 72711722 IC50 = 2800 nM T37848 C4O2MG 72711724 IC50 = 1600 nM T37848 C7PH3X 72711926 IC50 = 1900 nM T37848 C6NOU0 72711928 IC50 = 2300 nM T37848 CY4F2O 72711930 IC50 = 3200 nM T37848 CJM96S 72711932 IC50 = 10000 nM T37848 CQ72YG 72712127 IC50 = 4800 nM T37848 C3UF4Z 72712129 IC50 = 1700 nM T37848 C8WCQ4 72712131 Ki = 7100 nM T37848 C97PKX 72712133 Ki = 8500 nM T37848 CXLI39 72712342 Ki = 2100 nM T37848 CP5NK4 72712344 IC50 > 50000 nM T37848 C06CSU 72712346 IC50 = 37000 nM T37848 CBL6M3 72712570 Ki = 50000 nM T37848 CTQ42C 72712572 Ki = 50000 nM T37848 CE37QK 72713171 Ki = 1000 nM T37848 CLZ82F 72713536 IC50 = 48000 nM T37848 CHD69M 72713610 IC50 = 1300 nM T37848 CJA8Q5 72713752 IC50 > 50000 nM T37848 C7A5EW 72714054 IC50 = 18000 nM T37848 C7SZ3V 72714058 IC50 = 16000 nM T37848 C24PBI 72714290 IC50 = 1800 nM T37848 C3J0ZB 72725671 IC50 = 170 nM T37848 C8QEJ3 72725792 IC50 > 50000 nM T37848 CGM10E 72737641 IC50 > 25000 nM T37848 C7AO4X 72792633 IC50 > 50000 nM T37848 CLK7O4 72792692 IC50 > 50000 nM T37848 CBM7W0 72793032 IC50 = 6600 nM T37848 CNHI43 72793033 IC50 = 6800 nM T37848 C5E7IF 72793034 IC50 = 18000 nM T37848 CR4U6G 72793098 IC50 > 40000 nM T37848 CX38EH 72793099 IC50 > 40000 nM T37848 CNFA68 72793323 IC50 = 7000 nM T37848 CHW6N1 72793324 IC50 = 3400 nM T37848 C8G0MY 72793393 IC50 > 40000 nM T37848 C6R8DI 72943374 IC50 > 20000 nM T37848 C59QLH 72943630 IC50 = 310 nM T37848 CFG97I 72950095 IC50 > 15000 nM T37848 C9WU2M 72950813 IC50 > 100000 nM T37848 C1QMY5 73053248 IC50 > 10000 nM T37848 CH1JK9 73213123 IC50 > 40000 nM T37848 CV6ZT3 73297271 IC50 > 27000 nM T37848 CLA35R 73332001 IC50 = 27000 nM T37848 C7B2VH 73332466 IC50 > 10000 nM T37848 CO7R8B 73347331 IC50 > 10000 nM T37848 CAV13P 73348835 IC50 > 30000 nM T37848 CFPW17 73348992 IC50 = 500 nM T37848 C57LGA 73349098 IC50 > 10000 nM T37848 CK40LM 73349243 IC50 = 900 nM T37848 CZ1V0X 73350418 IC50 > 10000 nM T37848 C80BSO 73352560 IC50 > 20000 nM T37848 C46KTL 73353391 IC50 > 30000 nM T37848 CG7R3F 73353420 IC50 > 30000 nM T37848 CM0W7S 73354069 IC50 > 20000 nM T37848 C3DJ5W 73356463 IC50 > 10000 nM T37848 C32YFH 73356464 IC50 > 30000 nM T37848 C6HBS9 73356465 IC50 > 10000 nM T37848 C0LF9I 73356861 IC50 > 10000 nM T37848 C9WY3B 73386689 Ki = 1640 nM T37848 CRA5H6 73389570 IC50 > 10000 nM T37848 C2PAK9 73438493 IC50 > 30000 nM T37848 CVF5P0 73603034 Ki = 1120 nM T37848 CDX9R1 73603344 IC50 > 50000 nM T37848 CTMF86 73603391 IC50 > 50000 nM T37848 C7LER5 73669500 IC50 > 50000 nM T37848 CJKB83 73670174 IC50 > 50000 nM T37848 CLZ7Q2 73670208 IC50 = 930 nM T37848 CHV3W1 73774630 IC50 > 30000 nM T37848 CYV4Z6 73890929 IC50 = 28000 nM T37848 CCFI76 73890932 IC50 = 960 nM T37848 C15QVF 74221424 IC50 = 5900 nM T37848 CZ3TB5 74221949 IC50 > 50000 nM T37848 CW9N8T 74222036 IC50 > 50000 nM T37848 CUF63H 74223858 IC50 > 30000 nM T37848 COE76R 74223859 IC50 > 30000 nM T37848 C7RAQ4 74538704 IC50 > 20000 nM T37848 C47JPV 75202872 IC50 = 800 nM T37848 C83YCN 75202873 IC50 = 19000 nM T37848 CPS18J 75276948 EC50 = 13000 nM T37848 C2G8VR 75593287 IC50 = 1630 nM T37848 CB4V1R 76071142 IC50 = 3200 nM T37848 CBAT06 76071144 IC50 > 30000 nM T37848 C7SH1T 76071506 IC50 = 1100 nM T37848 CS87EI 76071624 IC50 = 2400 nM T37848 C9E0PX 76071764 IC50 = 200 nM T37848 C1Y7HC 76072411 IC50 = 140 nM T37848 C0N3RW 76282073 IC50 > 20000 nM T37848 C20YHA 76283431 IC50 > 30000 nM T37848 CHV72I 76283681 IC50 > 20000 nM T37848 CT59ZA 76283684 IC50 > 20000 nM T37848 CE2NP9 76284760 IC50 > 20000 nM T37848 C5ALQ2 76285468 IC50 > 30000 nM T37848 CH89VC 76310149 IC50 = 16000 nM T37848 C7JAY2 76310561 IC50 = 240 nM T37848 CQY40K 76310562 IC50 = 220 nM T37848 C0AOG7 76310563 IC50 = 460 nM T37848 CA70YQ 76310589 IC50 > 30000 nM T37848 CF95ZW 76310603 IC50 = 120 nM T37848 CY0HD7 76311092 IC50 = 180 nM T37848 CAT65E 76311096 IC50 = 1200 nM T37848 CF07EK 76313382 IC50 > 20000 nM T37848 CMF40L 76313439 IC50 = 1100 nM T37848 C5EB1U 76313856 IC50 = 17000 nM T37848 C3SCB2 76314207 IC50 = 340 nM T37848 CI5M1J 76314237 IC50 = 130 nM T37848 CWH9N6 76314238 IC50 = 120 nM T37848 CQFG10 76314530 IC50 > 50000 nM T37848 CX3LZ0 76314702 IC50 = 65 nM T37848 CJO15N 76316894 IC50 > 20000 nM T37848 CK09EA 76317380 IC50 > 20000 nM T37848 C6Z1BP 76317768 IC50 = 440 nM T37848 CKN6O4 76317769 IC50 = 1100 nM T37848 C3OP2B 76319044 IC50 > 10000 nM T37848 CCMW30 76320680 IC50 > 50000 nM T37848 C9JAG2 76321101 IC50 = 7000 nM T37848 CR02UI 76321102 IC50 = 4000 nM T37848 CV8YN2 76321484 IC50 = 310 nM T37848 C5JOH3 76321485 IC50 = 1840 nM T37848 C86CEF 76321486 IC50 = 350 nM T37848 CN40LR 76321520 IC50 = 110 nM T37848 CEK3O5 76321713 IC50 > 30000 nM T37848 CNY2D6 76321910 EC50 = 14000 nM T37848 C7Y5QF 76321979 IC50 = 270 nM T37848 CR05PL 76322043 IC50 > 100000 nM T37848 CQ3CW1 76322044 IC50 = 41800 nM T37848 CYXU43 76322162 IC50 > 30000 nM T37848 CR7FP8 76324529 IC50 = 4500 nM T37848 CA1TW6 76324750 IC50 > 20000 nM T37848 CVTY04 76324753 IC50 = 12000 nM T37848 C5C8JD 76324755 IC50 > 20000 nM T37848 CH9NX4 76325091 IC50 = 1260 nM T37848 C2SM8Y 76325108 IC50 > 30000 nM T37848 C1HFI9 76325446 IC50 = 25000 nM T37848 C1HJQ9 76325597 IC50 = 1400 nM T37848 C3C7HE 76325645 IC50 = 2200 nM T37848 C2HCL6 76327886 IC50 > 50000 nM T37848 CYR3L4 76327922 IC50 = 44000 nM T37848 CQ39WV 76328292 IC50 = 6300 nM T37848 C5PW1E 76328299 IC50 = 5200 nM T37848 CD0KS8 76328654 IC50 = 630 nM T37848 CO6XN0 76328655 IC50 = 1670 nM T37848 CB3LV0 76328656 IC50 = 1400 nM T37848 CJ9N0S 76328675 IC50 > 30000 nM T37848 C5UMK8 76328829 IC50 > 30000 nM T37848 C8CQ9Y 76328873 IC50 > 30000 nM T37848 CZ9Q2S 76329164 IC50 = 2000 nM T37848 CWD5R4 76331595 IC50 = 25000 nM T37848 CB2VE0 76331988 IC50 > 20000 nM T37848 CE6BI0 76332666 IC50 = 40000 nM T37848 CZ2CQ7 76332826 IC50 = 2500 nM T37848 C76UKL 76333454 IC50 > 20000 nM T37848 CR4HY1 76335555 IC50 > 20000 nM T37848 C0TLY1 76335557 IC50 = 16000 nM T37848 C0JHC6 76335558 IC50 > 20000 nM T37848 CR2B8N 76335560 IC50 > 20000 nM T37848 CDM50P 76335564 IC50 = 18000 nM T37848 C9QYB2 76335964 IC50 = 140 nM T37848 CC9BJ5 76335965 IC50 = 300 nM T37848 CE4YP9 76335969 IC50 > 10000 nM T37848 CVUY84 76335992 IC50 = 80 nM T37848 CGE5S3 76336366 EC50 > 40000 nM T37848 CGJM01 76336447 IC50 > 10000 nM T37848 C92WBQ 76336500 IC50 = 86000 nM T37848 CAT95V 76685067 IC50 = 85120 nM T37848 C8CP3K 76903477 IC50 > 50000 nM T37848 CQT14W 76955651 IC50 > 30000 nM T37848 C7F2RD 77050711 IC50 = 65000 nM T37848 C34TAM 77845572 IC50 > 50000 nM T37848 C1YJW0 77846787 IC50 = 336 nM T37848 CV73PD 77846790 IC50 = 87 nM T37848 C0DIH7 77846872 IC50 = 145 nM T37848 COI25M 77846873 IC50 = 151 nM T37848 CJI8R0 77846875 IC50 = 99 nM T37848 CZK4J1 77846962 IC50 = 153 nM T37848 CEK89G 77846963 IC50 = 185 nM T37848 C5BA8Z 77846964 IC50 = 226 nM T37848 C4D6XJ 77847803 IC50 = 162 nM T37848 CF7O4Q 77847804 IC50 = 198 nM T37848 CWG4T2 78209992 IC50 > 50 nM T37848 C2NCH9 78318214 IC50 > 50000 nM T37848 C2GET7 78318815 IC50 > 50000 nM T37848 CLB1A4 78319901 IC50 > 50000 nM T37848 C9GQS2 81689815 IC50 > 100000 nM T37848 C3H5XR 82639722 IC50 > 10000 nM T37848 CQMB31 85470872 IC50 = 2300 nM T37848 C15BSO 86270136 IC50 > 10000 nM T37848 CA1CE3 86270720 IC50 = 2000 nM T37848 CXN93A 86271108 IC50 > 10000 nM T37848 C2KHM0 86271111 IC50 > 10000 nM T37848 CZL23E 86271138 IC50 > 30000 nM T37848 C5IR2K 86271238 IC50 > 30000 nM T37848 CN9MO7 86271494 IC50 > 10000 nM T37848 C4T3IW 86272102 IC50 > 100000 nM T37848 C13AJC 86274362 IC50 = 63000 nM T37848 C3OLB1 86274489 IC50 > 100000 nM T37848 CAB78T 86274732 IC50 > 100000 nM T37848 CCU13T 86275207 IC50 = 31000 nM T37848 CJ68CO 86275449 IC50 > 100000 nM T37848 CF4QX9 86278359 IC50 > 10000 nM T37848 CXF9Q3 86279146 IC50 = 9400 nM T37848 C4Y3VP 86279147 IC50 = 20000 nM T37848 CPJV10 86280878 IC50 > 10000 nM T37848 CYK2T9 86282366 IC50 = 3300 nM T37848 CH3FN8 86288905 IC50 = 12000 nM T37848 CKQ71X 86288935 IC50 = 19540 nM T37848 C36LAF 86302354 IC50 = 25000 nM T37848 CMKO61 86303027 IC50 > 20000 nM T37848 C3Y9KN 86303187 IC50 = 5200 nM T37848 C6A1DG 86304283 IC50 < 46 nM T37848 C0IZU4 86304284 IC50 = 8000 nM T37848 C5JFM1 86304285 IC50 = 53000 nM T37848 CKJI10 86304439 IC50 = 50000 nM T37848 CGK31H 86304440 IC50 = 42000 nM T37848 CJ7SI6 86304441 IC50 > 100000 nM T37848 C9EMQ0 86304601 IC50 > 34000 nM T37848 CV4Q5D 86304762 IC50 = 12000 nM T37848 CB5F1W 86343364 IC50 > 30000 nM T37848 CKG7N2 86343365 IC50 > 30000 nM T37848 C9IVM5 86343366 IC50 > 30000 nM T37848 CK02ZT 86344136 IC50 = 32000 nM T37848 CZU43C 86344330 IC50 = 3600 nM T37848 C6D5QL 86344510 IC50 > 50000 nM T37848 CMG39E 86673884 IC50 = 17000 nM T37848 CTG76E 86687532 IC50 > 50000 nM T37848 CFT89Y 86687602 IC50 > 27000 nM T37848 CY8JW3 86687604 IC50 > 27000 nM T37848 C7OXV8 86687606 IC50 > 27000 nM T37848 C47MVU 86695644 IC50 = 6900 nM T37848 CC8I0M 86707711 IC50 = 11000 nM T37848 COW7F1 86711021 IC50 = 1500 nM T37848 C53FOY 86711045 IC50 = 1500 nM T37848 CVJ8L5 86728666 IC50 = 50 nM T37848 CQ45XR 86763358 IC50 > 15848.93 nM T37848 CTW8L6 86766622 IC50 = 3800 nM T37848 C2U0BG 87055263 IC50 > 10000 nM T37848 CG0U7A 87451692 IC50 = 100 nM T37848 C0Y1VJ 87451777 IC50 = 1200 nM T37848 CSRU90 87550393 IC50 = 1900 nM T37848 CF67AV 88875879 IC50 = 16000 nM T37848 C8Y9RW 89462922 IC50 > 12.5 nM T37848 C0DRH8 89463724 IC50 = 2.4 nM T37848 C8SK1N 89463725 IC50 > 12.5 nM T37848 CL30TR 89471870 IC50 > 25000 nM T37848 C3BUS8 89471889 IC50 = 11000 nM T37848 CI7HY8 89471890 IC50 = 2800 nM T37848 C8OSN4 89509786 IC50 = 1000 nM T37848 CR0P6K 89584034 IC50 > 50000 nM T37848 CM6SL8 89613863 IC50 = 7200 nM T37848 C90UQK 89614650 IC50 = 1300 nM T37848 CYK8P4 89619265 IC50 > 200000 nM T37848 CR8P9M 89619268 IC50 > 200000 nM T37848 CNU89Y 89619334 IC50 > 200000 nM T37848 CGC40J 89619484 IC50 > 200000 nM T37848 C93RQC 89619504 IC50 > 200000 nM T37848 C1HE4A 89619588 IC50 = 10000 nM T37848 C7MNP5 89619702 IC50 = 122000 nM T37848 C6T4OW 89634586 IC50 > 200000 nM T37848 CA49UY 89726151 IC50 > 30000 nM T37848 CY6K5P 89738540 IC50 > 30000 nM T37848 CIXB02 89738547 IC50 = 14200 nM T37848 CG9CM0 89750383 IC50 = 11000 nM T37848 C2BM9L 89768534 IC50 > 30000 nM T37848 CB4Y7R 89768546 IC50 > 30000 nM T37848 C5MR9K 89777151 IC50 > 30000 nM T37848 CRZ34V 89777258 IC50 = 340 nM T37848 CZ58KT 89777437 IC50 = 25000 nM T37848 C5S4PX 89777463 IC50 = 24000 nM T37848 CI57QV 89782019 IC50 > 50000 nM T37848 CK9I5Y 89789751 IC50 = 8800 nM T37848 C9I6NQ 89789762 IC50 > 50000 nM T37848 C8S7BC 89789778 IC50 = 21000 nM T37848 CERC67 89789843 IC50 = 18000 nM T37848 CUS70D 89793496 IC50 > 10000 nM T37848 CP7MZ2 89793516 IC50 > 10000 nM T37848 C9X5OT 89793519 IC50 > 10000 nM T37848 C96EWN 89795484 IC50 > 10000 nM T37848 CWO58S 89795501 IC50 > 10000 nM T37848 CIQ53M 89795553 IC50 > 10000 nM T37848 C5GQL0 89795796 IC50 > 10000 nM T37848 CGD0S5 89825760 IC50 = 3900 nM T37848 CA34IP 89826402 IC50 > 50000 nM T37848 C7GC8K 89826796 IC50 > 20000 nM T37848 C1IA0Q 89826982 IC50 > 20000 nM T37848 CMJY71 89827041 IC50 > 20000 nM T37848 CT6W0Y 89835558 IC50 = 5600 nM T37848 C16AXO 89846366 IC50 > 50000 nM T37848 CEK2I7 89846957 IC50 > 20000 nM T37848 C4MJ6O 89846958 IC50 > 50000 nM T37848 CMS6X4 89931025 IC50 = 1400 nM T37848 CX0M7B 89961716 IC50 = 36510 nM T37848 C7CQD4 89971933 IC50 = 2400 nM T37848 CQ5HZ7 89996234 IC50 > 50000 nM T37848 CI54WQ 89996408 IC50 > 15000 nM T37848 CJ65EF 90012001 IC50 > 10000 nM T37848 CW7R5J 90112663 IC50 = 3100 nM T37848 C18EVT 90130762 IC50 = 3000 nM T37848 CGN3K4 90130771 IC50 = 5000 nM T37848 COVK20 90142631 IC50 > 40000 nM T37848 C3YPA8 90149424 IC50 = 1900 nM T37848 C1Q6PT 90149477 IC50 > 30000 nM T37848 C63ZAP 90176119 IC50 > 20000 nM T37848 CY5IC7 90252834 IC50 = 43000 nM T37848 C84NVA 90252850 IC50 > 50000 nM T37848 CBY46O 90252851 IC50 > 50000 nM T37848 CNVA50 90252852 IC50 > 50000 nM T37848 CRN8G1 90253396 IC50 > 20000 nM T37848 C89BFG 90333640 IC50 = 185 nM T37848 C26LKW 90341025 IC50 > 50000 nM T37848 CE2XU8 90354304 IC50 = 1200 nM T37848 CE4IT5 90408860 IC50 > 10000 nM T37848 CB0RP3 90410604 IC50 > 10000 nM T37848 CQ8ZW3 90410911 IC50 > 10000 nM T37848 CD5W6K 90417914 IC50 = 43000 nM T37848 CJE7P5 90467013 IC50 > 50000 nM T37848 CX6DQ4 90467014 IC50 > 50000 nM T37848 C7D2UK 90467156 IC50 > 50000 nM T37848 CV75ZC 90467159 IC50 > 50000 nM T37848 C3RO1M 90467162 IC50 > 50000 nM T37848 C6BID5 90469437 IC50 > 10000 nM T37848 CF30KA 90643570 IC50 > 100000 nM T37848 CGS36U 90644505 IC50 = 216 nM T37848 CYE3G5 90644506 IC50 = 44.4 nM T37848 CDE57X 90644507 IC50 = 1080 nM T37848 CV53YI 90644508 IC50 = 1250 nM T37848 C1S8PM 90644647 IC50 = 7500 nM T37848 C5WDB0 90644648 IC50 = 900 nM T37848 C5O8HN 90644762 IC50 > 30000 nM T37848 CY4PB3 90644766 IC50 > 30000 nM T37848 CL5UB3 90644769 IC50 = 20300 nM T37848 C6AMK9 90644770 IC50 = 2400 nM T37848 CAVN86 90644773 IC50 = 14100 nM T37848 CEZK64 90645309 IC50 > 20000 nM T37848 CXUH46 90645310 IC50 > 20000 nM T37848 C0NM1C 90645311 IC50 = 1900 nM T37848 CL0O7Q 90645312 IC50 > 20000 nM T37848 C8YE0S 90654338 IC50 = 4000 nM T37848 C6AU0Q 90654563 IC50 = 400 nM T37848 CSW57N 90654564 IC50 = 2200 nM T37848 CY8VB0 90654565 IC50 = 700 nM T37848 CK8J1R 90654566 IC50 = 3000 nM T37848 C7R8YB 90654567 IC50 = 800 nM T37848 C23TZB 90654568 IC50 = 7800 nM T37848 C0KAP2 90654583 IC50 > 25000 nM T37848 CY8CN2 90654584 IC50 = 2000 nM T37848 CN8Y1A 90654585 IC50 = 7600 nM T37848 C0XQB9 90654586 IC50 > 25000 nM T37848 CHP74S 90654587 IC50 < 1000 nM T37848 C12FTL 90654588 IC50 < 100 nM T37848 CYXW14 90654589 IC50 = 1100 nM T37848 CPG7U1 90654590 IC50 = 10000 nM T37848 CMB8C2 90654591 IC50 < 300 nM T37848 CLME72 90654592 IC50 = 5200 nM T37848 C96YCU 90654600 IC50 > 25000 nM T37848 CV09GW 90655372 IC50 > 27000 nM T37848 CB2RM8 90655373 IC50 > 27000 nM T37848 CHBG56 90655374 IC50 = 2500 nM T37848 C0NXS3 90655376 IC50 = 3800 nM T37848 CV72RT 90655377 IC50 > 27000 nM T37848 CF68GW 90655378 IC50 = 700 nM T37848 CNBZ28 90655379 IC50 = 1300 nM T37848 C26LUH 90655380 IC50 = 500 nM T37848 CZD14Q 90655381 IC50 > 27000 nM T37848 C4OCF1 90655382 IC50 > 27000 nM T37848 COBZ93 90655383 IC50 = 700 nM T37848 CT4ZL3 90655384 IC50 = 1700 nM T37848 COZS39 90655385 IC50 = 800 nM T37848 CX6Z2P 90656800 IC50 = 4500 nM T37848 CMO7T8 90656801 IC50 = 6500 nM T37848 CE8OH5 90656802 IC50 = 27000 nM T37848 CI6P0E 90656803 IC50 = 1800 nM T37848 C5GA9J 90656804 IC50 = 9400 nM T37848 CL7PU4 90656805 IC50 = 100000 nM T37848 C0YK1U 90656806 IC50 = 25000 nM T37848 CWE0X5 90656807 IC50 = 81000 nM T37848 CIL2W9 90664452 IC50 > 20000 nM T37848 CSDO81 90664458 IC50 = 2730 nM T37848 CQT69X 90664721 IC50 > 100000 nM T37848 CN3A1P 90664848 IC50 > 100000 nM T37848 CJ01LW 90664969 IC50 > 100000 nM T37848 C01UNB 90665166 IC50 > 10000 nM T37848 CG98QO 90665194 IC50 > 20000 nM T37848 C02PLA 90665208 IC50 > 100000 nM T37848 CG4E8W 90665845 IC50 = 680 nM T37848 CXEJ32 90665986 IC50 = 5400 nM T37848 CDQ56W 90665987 IC50 = 13700 nM T37848 C5E2FJ 90665988 IC50 > 30000 nM T37848 CXEK45 90681222 IC50 = 300 nM T37848 C8H4KE 90681223 IC50 < 300 nM T37848 CA9PL8 91663316 IC50 > 30000 nM T37848 CQS8C9 91664365 IC50 = 9360 nM T37848 C65ANP 91666625 IC50 = 38800 nM T37848 C26BZK 91666633 IC50 > 10000 nM T37848 C9ETC1 91666645 IC50 > 50000 nM T37848 CUI10E 91666686 IC50 > 30000 nM T37848 C2H7XV 91668260 IC50 > 5000 nM T37848 C4YP6M 91754658 IC50 = 6800 nM T37848 C5CKD3 91754690 IC50 > 20000 nM T37848 CM95VC 91758806 IC50 = 260 nM T37848 C5T0FH 91799687 IC50 > 10000 nM T37848 CUX4B6 91809187 IC50 > 60000 nM T37848 CUQ1W0 91810395 IC50 = 13300 nM T37848 CK6E0W 91810397 IC50 = 2100 nM T37848 CWTO83 91810751 IC50 > 10000 nM T37848 CC9B6T 91820646 IC50 > 18000 nM T37848 C3L6KU 91820689 IC50 > 25000 nM T37848 C64QCZ 91827500 IC50 = 10000 nM T37848 CLB2E7 91827654 IC50 > 50000 nM T37848 CL7S4U 91844670 IC50 > 10000 nM T37848 C1JPD6 91844700 IC50 > 10000 nM T37848 CSK6Z1 91844707 IC50 > 10000 nM T37848 CH4L7O 91885483 IC50 > 30000 nM T37848 CBG6E7 91885506 IC50 > 5600 nM T37848 C75MDP 91885508 IC50 = 75000 nM T37848 CJ0P8X 91885509 IC50 = 520 nM T37848 CHTY48 91885510 IC50 = 210 nM T37848 C60HAJ 91885643 IC50 = 17000 nM T37848 CF8W2B 91928421 IC50 = 2100 nM T37848 CU1G3S 91933941 IC50 > 10000 nM T37848 C1SAH3 91971253 IC50 = 95000 nM T37848 CWZX73 91971958 IC50 >= 20000 nM T37848 CYMH49 92044895 IC50 = 29000 nM T37848 C57QJY 92045044 EC50 = 976 nM T37848 C38ZID 92045057 IC50 > 10000 nM T37848 CM6VG1 92239323 IC50 = 3200 nM T37848 CY2UI5 101891769 IC50 = 10100 nM T37848 CGB54P 101902999 IC50 = 4000 nM T37848 CG62HP 101903000 IC50 = 2900 nM T37848 C87GEW 102435977 IC50 > 10000 nM T37848 CQ9PN8 102593934 IC50 > 30000 nM T37848 C4Z1OU 110451319 IC50 = 10000 nM T37848 CN57AX 110451673 IC50 > 25000 nM T37848 CYX7T2 117072549 IC50 > 50000 nM T37848 C8F6VO 117604931 IC50 = 90000 nM T37848 CNFW42 117608566 IC50 > 10000 nM T37848 CGL3R6 117614609 IC50 = 1100 nM T37848 C6UOT8 117653759 IC50 > 20000 nM T37848 CL5OI9 117668598 IC50 > 20000 nM T37848 C5IO0K 117671078 IC50 > 20000 nM T37848 CE8SK5 117671214 IC50 > 20000 nM T37848 CVI38D 117737118 IC50 > 50000 nM T37848 CS4IW2 117739617 IC50 > 50000 nM T37848 C4ZO0A 117741876 IC50 > 27000 nM T37848 CBL12U 117748926 IC50 = 45000 nM T37848 C10BKY 117749324 IC50 > 50000 nM T37848 CQ2C1F 117751256 IC50 = 240 nM T37848 C4QN9K 117751334 IC50 = 60 nM T37848 CHQJ26 117751337 IC50 = 360 nM T37848 CS2A6Q 117751339 IC50 = 1400 nM T37848 C6XC3W 117769575 IC50 = 3000 nM T37848 CS72RV 117885758 IC50 > 50000 nM T37848 C6Z3NJ 117885766 IC50 > 50000 nM T37848 CKU6S4 117885912 IC50 > 50000 nM T37848 C89EQN 117897570 IC50 > 7200 nM T37848 CNS91H 117909194 IC50 = 50000 nM T37848 CR07ZG 117909666 IC50 = 21800 nM T37848 C6N8SM 117909768 IC50 = 9900 nM T37848 C9KV7L 117993993 IC50 > 50000 nM T37848 CNV24M 117993998 IC50 = 48600 nM T37848 CGBO72 118016229 IC50 > 20000 nM T37848 CJB47R 118086034 IC50 = 510 nM T37848 C3TBD8 118103460 IC50 > 30000 nM T37848 CZR2Q1 118103881 IC50 = 2300 nM T37848 CL15XC 118103886 IC50 = 2100 nM T37848 CI9Q2H 118103892 IC50 = 2000 nM T37848 CI3KM2 118103909 IC50 = 23000 nM T37848 CAIU03 118104096 IC50 = 10600 nM T37848 CIL65X 118104099 IC50 = 1900 nM T37848 CMX3U8 118107483 IC50 >= 5000 nM T37848 CWR6I1 118112300 IC50 > 20000 nM T37848 CNM1W9 118141977 IC50 = 8340 nM T37848 C56INY 118142016 IC50 = 38000 nM T37848 CN1LC9 118142017 IC50 = 30800 nM T37848 CZ0E5W 118142030 IC50 > 50000 nM T37848 CW5N0O 118142047 IC50 = 15500 nM T37848 CWL5J8 118174040 IC50 = 8000 nM T37848 CS6Y1X 118174075 IC50 > 30000 nM T37848 CF38UC 118174137 IC50 = 6200 nM T37848 CKXC27 118174156 IC50 = 5200 nM T37848 CDA16S 118174232 IC50 = 16000 nM T37848 CS7ER1 118174312 IC50 = 7100 nM T37848 CR4DE7 118175009 IC50 > 10000 nM T37848 C2U3TJ 118208018 IC50 > 20000 nM T37848 C6HSC3 118217854 IC50 > 10000 nM T37848 CEKH57 118217858 IC50 > 10000 nM T37848 CRM37Z 118223719 IC50 = 3500 nM T37848 CEN18L 118224069 IC50 = 22200 nM T37848 CT42ZR 118261815 IC50 > 50000 nM T37848 C3R9TY 118324047 IC50 > 10000 nM T37848 C7AO1M 118324066 IC50 > 10000 nM T37848 CPO08K 118344339 IC50 > 20000 nM T37848 CTCQ02 118344344 IC50 = 16000 nM T37848 C1HX3A 118344346 IC50 > 20000 nM T37848 CI7P6J 118344348 IC50 > 20000 nM T37848 C8J1PY 118344351 IC50 > 20000 nM T37848 CAWZ16 118344383 IC50 > 20000 nM T37848 CSUK24 118344385 IC50 = 18000 nM T37848 CA1YM6 118344504 IC50 > 20000 nM T37848 CC3N6Z 118344616 IC50 > 20000 nM T37848 CC0RD7 118345442 IC50 > 20000 nM T37848 CK43EA 118345549 IC50 = 19000 nM T37848 C0MCW3 118346170 IC50 > 20000 nM T37848 CRZ5N1 118368912 IC50 > 50000 nM T37848 CBIR89 118389918 IC50 = 16300 nM T37848 CY0K6A 118452766 IC50 = 780 nM T37848 C86XOE 118452846 IC50 = 3000 nM T37848 CR7DJ0 118453722 IC50 > 50000 nM T37848 CK1Z7I 118462026 IC50 > 50000 nM T37848 CM2NH5 118478848 IC50 = 11000 nM T37848 CRV8S3 118478927 IC50 > 10000 nM T37848 CL32JE 118478933 IC50 > 10000 nM T37848 C5S1HZ 118478972 IC50 > 10000 nM T37848 C8G9HP 118478986 IC50 > 10000 nM T37848 CBV89G 118478994 IC50 > 10000 nM T37848 CK0ER5 118478999 IC50 > 10000 nM T37848 CU25KC 118479000 IC50 > 10000 nM T37848 CW07IS 118479006 IC50 > 10000 nM T37848 C3ZAV0 118479034 IC50 > 10000 nM T37848 C4W6ZS 118479038 IC50 > 10000 nM T37848 CRG24C 118479053 IC50 > 10000 nM T37848 CD4ME1 118479123 IC50 > 10000 nM T37848 CB0XM2 118479161 IC50 > 10000 nM T37848 C18NTQ 118479199 IC50 > 10000 nM T37848 CJ0Z1Y 118479222 IC50 > 10000 nM T37848 CP0U6Y 118479229 IC50 > 10000 nM T37848 C3A6HD 118479231 IC50 > 10000 nM T37848 CJ14CR 118479241 IC50 > 10000 nM T37848 C1FO3N 118479293 IC50 > 10000 nM T37848 CF02TZ 118479295 IC50 > 10000 nM T37848 C90TED 118479305 IC50 > 10000 nM T37848 C7I9RC 118479316 IC50 > 10000 nM T37848 CRC4F6 118479354 IC50 > 10000 nM T37848 CRCV51 118479359 IC50 > 10000 nM T37848 CJL5W0 118479428 IC50 > 10000 nM T37848 CS2VA7 118479440 IC50 > 10000 nM T37848 CJ9P0M 118479445 IC50 > 10000 nM T37848 C3U1RB 118479452 IC50 > 10000 nM T37848 CBJ28X 118483320 IC50 = 74000 nM T37848 C8PU5O 118491249 IC50 > 10000 nM T37848 C3KAO6 118491258 IC50 > 20000 nM T37848 CINA28 118492166 IC50 = 26000 nM T37848 CJ9Z0S 118496546 IC50 > 50000 nM T37848 C7AYV5 118540795 IC50 = 1150 nM T37848 CB41MH 118560618 IC50 = 46000 nM T37848 C78LNX 118572065 IC50 > 30000 nM T37848 CM93VO 118611725 IC50 > 20000 nM T37848 C0XJT5 118626089 IC50 = 10000 nM T37848 CRS34C 118705500 IC50 > 100000 nM T37848 C2LOB4 118706405 IC50 = 7000 nM T37848 CLUN23 118706414 IC50 > 20000 nM T37848 C2BG1F 118706537 IC50 = 600 nM T37848 C2WP6X 118706538 IC50 = 710 nM T37848 CZE4U0 118706539 IC50 = 510 nM T37848 CX8I0G 118706540 IC50 = 400 nM T37848 C18OLB 118706953 IC50 = 46000 nM T37848 CS7HY2 118707102 IC50 = 36000 nM T37848 CTM4S1 118707103 IC50 = 54000 nM T37848 CS4R3B 118707826 IC50 > 30000 nM T37848 CLS7C1 118707978 IC50 > 40000 nM T37848 C9LV0M 118707979 IC50 = 300 nM T37848 CR8VJ2 118708873 IC50 > 5000 nM T37848 CL2VY5 118708881 IC50 > 5000 nM T37848 CB5F2O 118708929 IC50 > 5000 nM T37848 C8M3JX 118708934 IC50 > 5000 nM T37848 C9W3LI 118708938 IC50 > 5000 nM T37848 CEAK31 118708939 IC50 > 5000 nM T37848 CMX6S5 118709259 IC50 > 20000 nM T37848 CG19YT 118709623 IC50 = 27000 nM T37848 CT1J7Y 118709777 IC50 = 270 nM T37848 CT91SV 118711722 IC50 > 20000 nM T37848 C4T2FY 118712775 IC50 = 56490 nM T37848 C5M3BX 118712788 IC50 = 2250 nM T37848 C4VAE0 118713757 IC50 = 1330 nM T37848 C84GOU 118713773 IC50 = 500 nM T37848 C2LY9D 118713799 IC50 = 32700 nM T37848 CMO2V7 118713801 IC50 = 1100 nM T37848 C9LKI0 118713803 IC50 = 810 nM T37848 C2OZ7H 118713805 IC50 = 3640 nM T37848 CM4P8X 118713806 IC50 = 500 nM T37848 C7EXQ9 118713807 IC50 = 120 nM T37848 CUM74B 118716060 IC50 > 10000 nM T37848 CLGD29 118720097 IC50 = 6710 nM T37848 C4LW6I 118720885 IC50 > 40000 nM T37848 C9SF2E 118720891 IC50 > 24000 nM T37848 C6Y5JG 118723171 IC50 = 2000 nM T37848 CE3I9T 118723172 IC50 = 4000 nM T37848 C13AIC 118723173 IC50 = 500 nM T37848 C21SWI 118723174 IC50 = 2000 nM T37848 CKR24J 118723175 IC50 = 700 nM T37848 C28YZF 118723176 IC50 = 2000 nM T37848 C4QO8E 118723178 IC50 = 2000 nM T37848 C2EH1G 118723182 IC50 = 51000 nM T37848 C3R7XB 118725448 IC50 = 1000 nM T37848 CT4WP3 118725451 IC50 > 10000 nM T37848 C3SAQ6 118725452 IC50 > 10000 nM T37848 CQ6HI7 118725453 IC50 > 10000 nM T37848 CS1FU0 118725519 IC50 = 4500 nM T37848 C3QD8O 118725520 IC50 = 50 nM T37848 C6LWF1 118725521 IC50 = 490 nM T37848 CO30HX 118725522 IC50 = 80 nM T37848 CR95GT 118725524 IC50 = 500 nM T37848 C6RXB2 118729222 IC50 > 40000 nM T37848 C9HFE1 118730345 IC50 > 10000 nM T37848 C6HV3B 118730351 IC50 > 10000 nM T37848 C3LZM9 118730352 IC50 > 7000 nM T37848 CTE58Z 118730369 IC50 = 2500 nM T37848 C1PR2Q 118730373 IC50 = 70000 nM T37848 C52QGJ 118730382 IC50 = 900 nM T37848 C4EI0W 118730384 IC50 = 300 nM T37848 C6B4XD 118730937 IC50 > 20000 nM T37848 CO81CK 118730940 IC50 > 20000 nM T37848 C27FIO 118730943 IC50 > 20000 nM T37848 CLU74Q 118731287 IC50 = 450 nM T37848 C65YAM 118731484 IC50 = 23500 nM T37848 C4YQN5 118731487 IC50 = 21700 nM T37848 CC3PT6 118731957 IC50 = 46000 nM T37848 C7R8HJ 118732962 IC50 > 50000 nM T37848 C6OEU2 118733374 IC50 > 50000 nM T37848 C4G3YC 118734875 IC50 > 30000 nM T37848 C9AIE1 118734876 IC50 > 30000 nM T37848 CAN90V 118735353 IC50 = 2000 nM T37848 C4XY9I 118735354 IC50 > 100000 nM T37848 C1XL4S 118735355 IC50 = 35000 nM T37848 CQSF74 118735386 IC50 = 410 nM T37848 C2P7NL 118735389 IC50 = 2100 nM T37848 CB57VC 118737720 IC50 > 50000 nM T37848 C15QMA 118737724 IC50 > 50000 nM T37848 C1MHT0 118737725 IC50 > 50000 nM T37848 C5BOQ1 118753201 Ki > 30000 nM T37848 C87ZPY 118796358 IC50 > 50000 nM T37848 CIPQ86 118861736 EC50 = 1030 nM T37848 CR71BE 118861737 EC50 = 4640 nM T37848 CDSY04 118861738 EC50 = 2460 nM T37848 C9WBY6 118861778 EC50 = 3990 nM T37848 CELZ36 118866105 IC50 = 27000 nM T37848 C14DLY 118872292 IC50 = 50000 nM T37848 CM59EQ 118917669 IC50 > 30000 nM T37848 C6J8YF 118917671 IC50 = 620 nM T37848 C2RBF7 118918048 IC50 = 13000 nM T37848 CL4KX1 118950056 IC50 = 370 nM T37848 CC4LA1 118953461 IC50 > 30000 nM T37848 C8L1QI 118959080 IC50 > 5000 nM T37848 C9LR8Z 118965395 IC50 > 100000 nM T37848 C13EIL 118967091 IC50 = 14000 nM T37848 CE3CN6 118971057 IC50 = 17600 nM T37848 C4K3PR 118987036 IC50 > 25000 nM T37848 COS3K9 121304408 IC50 > 5000 nM T37848 C9G3ZJ 121304414 IC50 > 7000 nM T37848 C4RD9Y 121304424 IC50 > 17000 nM T37848 C1PKR0 121304441 IC50 > 3000 nM T37848 CC3MP6 121304452 IC50 > 3000 nM T37848 CW68KD 121304458 IC50 > 50000 nM T37848 CPB58L 121304467 IC50 > 9000 nM T37848 COB2X5 121304477 IC50 > 2000 nM T37848 CZ0BI4 121304484 IC50 > 38000 nM T37848 CW51NQ 121304485 IC50 = 300 nM T37848 CX1DQ6 121304488 IC50 > 6000 nM T37848 C7NLV2 121304500 IC50 > 10000 nM T37848 CQ2UM4 121304538 IC50 > 17000 nM T37848 C1AB6P 121304551 IC50 = 3400 nM T37848 CN05ZQ 121304574 IC50 > 17000 nM T37848 CU0M7B 121304590 IC50 > 17000 nM T37848 CX5MO3 121304598 IC50 > 6000 nM T37848 C2VTK5 121304654 IC50 > 10000 nM T37848 C6IB0P 121304685 IC50 > 21000 nM T37848 CXC70Q 121304711 IC50 > 7000 nM T37848 C6C9EF 121304827 IC50 = 2164 nM T37848 CU4CW1 121313969 IC50 > 50000 nM T37848 C65ZYO 121332604 IC50 > 3000 nM T37848 C92NOH 121332654 IC50 > 3000 nM T37848 CNBH32 121332727 IC50 > 3000 nM T37848 C9H0BR 121333853 IC50 > 27000 nM T37848 C83STC 121333902 IC50 > 27000 nM T37848 CMA2O3 121333930 IC50 > 27000 nM T37848 C9Q2ND 121333973 IC50 > 15000 nM T37848 C6TBD2 121345502 IC50 > 50000 nM T37848 C34RDH 121346173 IC50 = 12000 nM T37848 C4CPO3 121398401 IC50 > 25000 nM T37848 C59ORZ 121398668 IC50 > 10000 nM T37848 CV9TX1 121399281 IC50 > 50000 nM T37848 C2WD1Q 121407246 IC50 > 50000 nM T37848 C9CV7H 121411850 IC50 > 20000 nM T37848 CU3BI0 121412063 IC50 > 20000 nM T37848 CQZ9W3 121414283 IC50 > 25000 nM T37848 C91PVZ 121428416 IC50 > 10000 nM T37848 C3KNZ5 121439991 IC50 > 3500 nM T37848 CQD4P5 121469330 IC50 = 2400 nM T37848 CV5R4G 121470704 IC50 = 44700 nM T37848 C85HZL 121470706 IC50 = 13900 nM T37848 C09QGL 121470709 IC50 = 37000 nM T37848 CWI1Z8 121472067 IC50 = 7500 nM T37848 CT7YX5 121472072 IC50 = 30000 nM T37848 C3OL2H 121480641 IC50 = 27200 nM T37848 CD89ZC 121480642 IC50 > 50000 nM T37848 CHD26A 121596332 IC50 > 20000 nM T37848 C3RFZ1 121596966 IC50 = 3050 nM T37848 CP52DJ 121596967 IC50 = 15400 nM T37848 CL8GC2 122177113 IC50 > 10000 nM T37848 C0H8AW 122177723 IC50 = 6500 nM T37848 C9WB6E 122179416 IC50 = 932 nM T37848 CYFA75 122179419 IC50 = 2740 nM T37848 CNGQ19 122179477 IC50 > 10000 nM T37848 CHE12L 122185954 IC50 = 12589.25 nM T37848 CR9AX0 122185958 IC50 = 3981.07 nM T37848 CEV6S8 122185963 IC50 = 7943.28 nM T37848 CK0UN1 122185974 IC50 = 10000 nM T37848 CQ1WJ8 122185975 IC50 = 12589.25 nM T37848 C3ZNU8 122185980 IC50 = 3981.07 nM T37848 CQA8B2 122187067 IC50 > 100000 nM T37848 CS5CF1 122187069 IC50 > 100000 nM T37848 C14FGL 122187534 IC50 > 20000 nM T37848 CB7IJ0 122188138 IC50 > 20000 nM T37848 C9TF8M 122190433 IC50 > 30000 nM T37848 CCD9E8 122190697 IC50 = 1170 nM T37848 CF0KD5 122190700 IC50 = 4920 nM T37848 C8GHY3 122190972 IC50 > 30000 nM T37848 C2JN3R 122192148 IC50 > 10000 nM T37848 CTI2V5 122192293 IC50 > 40000 nM T37848 C4NUY0 122192382 IC50 > 10000 nM T37848 C1MVP5 122192989 IC50 = 33260 nM T37848 CLHV68 122192990 IC50 > 50000 nM T37848 C1N0HP 122193176 IC50 > 30000 nM T37848 CV8J6N 122193177 IC50 > 30000 nM T37848 CB8MH7 122193179 IC50 > 30000 nM T37848 CC6K9M 122193588 IC50 = 1200 nM T37848 CK8LM4 122193872 IC50 = 200 nM T37848 C6CN5X 122193876 IC50 = 314 nM T37848 CNJ3F4 122193877 IC50 = 263 nM T37848 CQX7P1 122195090 IC50 > 2000 nM T37848 CUE4R9 122195192 IC50 > 20000 nM T37848 CNF81V 122195193 IC50 > 20000 nM T37848 CCP5U2 122195692 IC50 > 30000 nM T37848 CCP15H 122197303 IC50 = 40 nM T37848 C1G3UQ 122197339 IC50 = 12000 nM T37848 C5JXL2 122199175 IC50 = 3700 nM T37848 CEX9B4 122199179 IC50 = 13800 nM T37848 C1T5SW 122199188 IC50 = 9100 nM T37848 C32PNV 122234475 IC50 > 20000 nM T37848 C1C9LI 122246967 IC50 = 4000 nM T37848 CGT12J 122419159 IC50 > 30000 nM T37848 CZ4U5A 122429808 IC50 > 39810.72 nM T37848 C0AKG9 122433571 IC50 = 6309.57 nM T37848 C15NCI 122439267 IC50 = 695 nM T37848 CX4T7L 122439274 IC50 = 243 nM T37848 CC2EZ8 122443959 IC50 > 20000 nM T37848 C2F6EH 122456006 IC50 > 30000 nM T37848 C6QHB4 122484585 IC50 = 23900 nM T37848 COX7E3 122510453 IC50 > 20000 nM T37848 CLM7K3 122604539 IC50 = 13300 nM T37848 C01JHI 122604566 IC50 = 6900 nM T37848 CU2K4P 122650372 IC50 = 6080 nM T37848 C3RCU4 122650378 IC50 = 350 nM T37848 CS47AD 122650581 IC50 = 2600 nM T37848 C85JKN 122668190 IC50 > 25000 nM T37848 CD6X5P 122669265 IC50 > 20000 nM T37848 C86VYP 122670110 IC50 > 30000 nM T37848 C1YK2E 122678192 IC50 > 20000 nM T37848 C4P9NG 122700657 EC50 = 89000 nM T37848 CU95PT 122707120 IC50 > 50000 nM T37848 CSLF20 123226629 IC50 > 30000 nM T37848 C7ZJ8U 123295297 IC50 > 30000 nM T37848 CT9K0V 124000588 IC50 > 10000 nM T37848 C6CA4O 124088406 IC50 = 33000 nM T37848 C5ZY7L 124114343 IC50 > 50000 nM T37848 CPO7N5 124125214 IC50 > 20000 nM T37848 C4VT3O 124127413 IC50 = 25000 nM T37848 CZEC76 124147932 IC50 > 50000 nM T37848 CEK31I 124148318 IC50 = 13000 nM T37848 C5H2QB 124150512 IC50 > 50000 nM T37848 C7TOU4 124175991 IC50 > 10000 nM T37848 C53AYP 124176028 IC50 > 10000 nM T37848 CL7K0C 124176200 IC50 > 10000 nM T37848 CYD04K 124176232 IC50 > 10000 nM T37848 CMS9P1 124176233 IC50 > 10000 nM T37848 C7EQH8 124176242 IC50 > 10000 nM T37848 CGJH79 124176281 IC50 > 10000 nM T37848 CCYK63 124176287 IC50 > 10000 nM T37848 CWF7N2 124176288 IC50 > 10000 nM T37848 CK0B3W 124176291 IC50 > 10000 nM T37848 CNC17W 124176295 IC50 > 10000 nM T37848 CMG02Z 124176321 IC50 > 10000 nM T37848 CQMU46 124201651 IC50 < 10000 nM T37848 CA3S8B 124221798 IC50 = 2800 nM T37848 C84FIJ 124221975 IC50 = 2200 nM T37848 CDS92J 126483508 IC50 > 50000 nM T37848 CP8W0X 126533801 IC50 > 1000 nM T37848 CIV7R0 126533969 IC50 > 17000 nM T37848 CI97TU 126533981 IC50 > 2000 nM T37848 CA4QM3 126534084 IC50 = 980 nM T37848 CIAD86 126534204 IC50 > 20000 nM T37848 C4R7XU 126534291 IC50 = 920 nM T37848 CVBX50 126534373 IC50 > 3000 nM T37848 CFA3D6 126534516 IC50 > 5000 nM T37848 C0WUJ5 126534771 IC50 > 1000 nM T37848 CX9LM7 126534859 IC50 > 15000 nM T37848 C6DLR7 126534986 IC50 > 1000 nM T37848 C9Q0VB 126535075 IC50 > 16000 nM T37848 CIZC84 126535109 IC50 > 25000 nM T37848 CTAG09 126567264 IC50 = 10900 nM T37848 C5QT4N 126567306 IC50 > 25000 nM T37848 C2LAM7 126591927 IC50 > 30000 nM T37848 COZ95K 126648919 IC50 = 60 nM T37848 CZ3TD0 126651203 IC50 > 50000 nM T37848 C0LTB9 126651349 IC50 > 50000 nM T37848 C5XF4M 126678836 IC50 = 1500 nM T37848 C1O5VB 126740610 IC50 = 17000 nM T37848 C9KEY6 126740618 IC50 = 23000 nM T37848 COE64S 126740626 IC50 = 46000 nM T37848 COF75Z 126970673 IC50 = 21000 nM T37848 CS1B2E 127020968 IC50 > 10000 nM T37848 CB2ZK5 127026165 IC50 > 30000 nM T37848 C7J5VX 127026166 IC50 > 30000 nM T37848 C9XU8I 127026167 IC50 > 30000 nM T37848 CU32KG 127026289 IC50 = 21940 nM T37848 CA42BO 127027101 IC50 > 30000 nM T37848 C09CHL 127027102 IC50 > 30000 nM T37848 CK2WV4 127028395 IC50 = 700 nM T37848 CZ72JM 127028414 IC50 = 300 nM T37848 C5FZ7T 127028415 IC50 = 300 nM T37848 CGR4U3 127028416 IC50 = 300 nM T37848 CH4M9N 127028417 IC50 = 300 nM T37848 C1R8JC 127028418 IC50 = 150 nM T37848 C8W7QS 127028419 IC50 > 13000 nM T37848 C1CWF9 127028424 IC50 = 2000 nM T37848 CQM96C 127028425 IC50 = 30 nM T37848 CU1CN2 127028426 IC50 = 200 nM T37848 C9R3XB 127028427 IC50 > 13000 nM T37848 CCK36V 127029882 IC50 = 4778 nM T37848 CVC84H 127029883 IC50 = 7040 nM T37848 CFY1P0 127029884 IC50 = 363 nM T37848 CU8Y7N 127030224 IC50 = 5544 nM T37848 CTEA14 127030225 IC50 = 6697 nM T37848 CLDC46 127031152 IC50 = 26139 nM T37848 C60SMC 127031153 IC50 = 25988 nM T37848 C0A5RC 127031270 IC50 > 50000 nM T37848 C5BJY6 127033009 IC50 = 4000 nM T37848 C2POU1 127033963 IC50 > 30000 nM T37848 C2JOP5 127034286 IC50 > 30000 nM T37848 CZ61LK 127034966 IC50 > 10000 nM T37848 CA0SN5 127034967 IC50 > 10000 nM T37848 CP0W4Y 127036068 IC50 > 30000 nM T37848 C0V4SJ 127036359 IC50 > 45000 nM T37848 CWDI07 127037076 IC50 > 20000 nM T37848 C8QIK9 127037551 IC50 > 50000 nM T37848 CZU7Q2 127037819 IC50 = 54300 nM T37848 C5VF7R 127037821 IC50 = 18900 nM T37848 C46ISV 127038222 IC50 = 7200 nM T37848 CI6HK4 127038465 IC50 = 18600 nM T37848 C9Y8VL 127038466 IC50 > 100000 nM T37848 CUBG78 127039139 IC50 > 50000 nM T37848 CLN20Q 127039167 IC50 = 25500 nM T37848 C3O7CA 127039374 IC50 = 44700 nM T37848 CA4ZB8 127039509 IC50 = 27300 nM T37848 C20VKF 127039824 IC50 = 41400 nM T37848 C60HOC 127040550 IC50 = 30000 nM T37848 C34BGK 127040715 IC50 > 30000 nM T37848 C0J8HC 127041348 IC50 > 3000 nM T37848 C7PU6F 127041479 IC50 = 27200 nM T37848 CCU4Z1 127041764 IC50 = 3910 nM T37848 CI5TA6 127041772 IC50 = 19500 nM T37848 C6HB0F 127041783 IC50 = 200 nM T37848 CQ1U5D 127041786 IC50 = 20000 nM T37848 CCJX69 127041842 IC50 > 20000 nM T37848 CS78AZ 127041951 IC50 > 30000 nM T37848 CU9C4S 127041952 IC50 > 6000 nM T37848 C63OPL 127042084 IC50 = 16300 nM T37848 CLY9S7 127043130 IC50 > 33000 nM T37848 CVRS53 127043426 IC50 > 30000 nM T37848 C24LTO 127043427 IC50 > 30000 nM T37848 CP42FD 127043428 IC50 > 30000 nM T37848 CM9E6H 127043474 IC50 > 33000 nM T37848 CP25DC 127043607 IC50 > 30000 nM T37848 CRD92M 127043853 IC50 > 33000 nM T37848 CC17ZV 127044314 IC50 > 33000 nM T37848 C40FHS 127044788 IC50 > 33000 nM T37848 CQCO27 127046038 IC50 > 30000 nM T37848 C34REM 127046317 IC50 > 30000 nM T37848 C9A1TG 127046557 IC50 > 30000 nM T37848 C57ZRE 127046727 IC50 > 50000 nM T37848 CH6W2T 127046982 IC50 = 1100 nM T37848 C7YML2 127047647 IC50 = 21100 nM T37848 CJH46E 127047680 IC50 < 1100 nM T37848 C48NCK 127047993 IC50 > 30000 nM T37848 C84TQV 127048530 IC50 > 20000 nM T37848 CX8W4F 127049041 IC50 = 470 nM T37848 CZV7Q0 127049047 IC50 > 10000 nM T37848 CB54VQ 127049048 IC50 > 10000 nM T37848 C9TUQ2 127049049 IC50 > 10000 nM T37848 CJ8SG3 127049204 IC50 > 50000 nM T37848 C7D5QM 127049475 IC50 > 10000 nM T37848 C3V9MD 127049476 IC50 > 10000 nM T37848 C2O5LX 127049804 IC50 = 22940 nM T37848 CUVQ34 127050762 IC50 > 50000 nM T37848 CS6C8O 127050851 IC50 = 4800 nM T37848 C1HAU4 127050852 IC50 > 10000 nM T37848 CLX8S5 127050856 IC50 > 10000 nM T37848 CJP90K 127051009 IC50 > 20000 nM T37848 C9V4EG 127051045 IC50 > 50000 nM T37848 CH46LU 127051126 IC50 = 500 nM T37848 C39WXP 127051127 IC50 = 300 nM T37848 C5J3KY 127051128 IC50 = 1000 nM T37848 C7E4QP 127051129 IC50 = 3800 nM T37848 C2QX0V 127051283 IC50 > 20000 nM T37848 C7KZJ2 127052145 IC50 = 19100 nM T37848 C38VGB 127052215 IC50 = 15500 nM T37848 CZO5C7 127052225 IC50 > 10000 nM T37848 COX90Y 127052226 IC50 > 10000 nM T37848 C7QG9O 127052430 IC50 = 30000 nM T37848 CK5GJ2 127052461 IC50 = 9300 nM T37848 CR7O3H 127052463 IC50 > 20000 nM T37848 C4CRE7 127052464 IC50 > 20000 nM T37848 C75EAL 127052638 IC50 > 50000 nM T37848 C2GY5W 127052655 IC50 = 19800 nM T37848 CPZ70S 127052897 Ki = 540 nM T37848 C5OE2H 127053611 IC50 > 20000 nM T37848 CN3XU0 127255875 IC50 > 30000 nM T37848 CEC17N 129164665 IC50 = 47000 nM T37848 CY4B7Z 129164668 IC50 > 50000 nM T37848 CAT90Y 129164701 IC50 = 8000 nM T37848 CUB58Q 129164743 IC50 > 50000 nM T37848 C81SHO 129178830 IC50 > 50000 nM T37848 CJGR20 129240126 IC50 > 30000 nM T37848 CP09TF 129282671 IC50 = 650 nM T37848 C42ZDX 129282689 IC50 = 600 nM T37848 C3GA7K 129282703 IC50 > 10000 nM T37848 CV28YE 129282706 IC50 = 2800 nM T37848 C3SGN0 129282870 IC50 = 2400 nM T37848 CU70NI 129282903 IC50 > 10000 nM T37848 C3CH6E 129283030 IC50 = 3300 nM T37848 C7FXS8 129283166 IC50 = 6000 nM T37848 C32WDC 129283174 IC50 = 840 nM T37848 C9HZ2S 129283211 IC50 = 8200 nM T37848 C5L7MR 129283737 IC50 > 10000 nM T37848 CE19JM 129296385 IC50 < 100 nM T37848 C7MRB5 129304758 IC50 = 2900 nM T37848 CE8TV5 129893260 IC50 < 10000 nM T37848 C9NPD3 129909153 IC50 > 25000 nM T37848 C4LR9M 129909326 IC50 > 25000 nM T37848 CD80OM 129909338 IC50 = 5920 nM T37848 CV3UP6 129909861 IC50 > 30000 nM T37848 CK68CA 130453737 IC50 > 30000 nM T37848 CDV84X 131747741 IC50 > 50000 nM T37848 CV06MU 131801402 IC50 = 1300 nM T37848 C4Z5MQ 131839619 IC50 > 30000 nM T37848 CFC05Q 131954513 IC50 > 30000 nM T37848 CN4RF6 132019596 IC50 > 30000 nM T37848 CZ5H2B 132020452 IC50 > 40000 nM T37848 CP8A1Q 132020575 IC50 = 15000 nM T37848 CH8DP7 132220479 IC50 > 20000 nM T37848 C5P4XN 132227197 IC50 > 18000 nM T37848 C1R5SZ 132227201 IC50 > 18000 nM T37848 CGDN94 132275066 IC50 > 10000 nM T37848 CF73XU 132473042 IC50 > 30000 nM T37848 C5U7JM 132473043 IC50 = 15000 nM T37848 CACJ46 132489333 IC50 > 25000 nM T37848 C6Z8BD 132510851 IC50 = 100 nM T37848 CN12VW 132550264 IC50 = 155 nM T37848 C9QYP1 132585220 IC50 = 16000 nM T37848 CJE34F 132597748 IC50 > 27000 nM T37848 CBXG19 132606863 IC50 = 1700 nM T37848 CYP29B 132990558 IC50 = 11200 nM T37848 C0AI1V 132991411 IC50 = 23 nM T37848 C39UCD 133080605 IC50 = 21000 nM T37848 CZC7S8 133081963 IC50 = 7730 nM T37848 C18GQC 134128280 IC50 > 20000 nM T37848 CY0GK7 134132068 IC50 = 18000 nM T37848 CO1RW6 134132142 IC50 = 3280 nM T37848 C9WK2U 134132312 IC50 > 30000 nM T37848 CL7WX2 134132313 IC50 = 2200 nM T37848 CZ8NM1 134133165 IC50 = 17000 nM T37848 CH7Q4E 134133267 IC50 > 50000 nM T37848 CW74SC 134133758 IC50 > 50000 nM T37848 CJOQ95 134134229 IC50 > 50000 nM T37848 CI8KY0 134135230 IC50 = 4000 nM T37848 CES87G 134135247 IC50 = 2500 nM T37848 CC7OQ2 134135307 IC50 > 50000 nM T37848 CLH5U3 134135450 IC50 = 15000 nM T37848 CE5TV4 134135453 IC50 = 15000 nM T37848 CGZ4Y6 134135730 IC50 = 8300 nM T37848 CDRC75 134136284 IC50 = 227 nM T37848 CK9MG1 134136380 IC50 = 18000 nM T37848 CHS48B 134137453 IC50 = 11000 nM T37848 C8K7CE 134138554 IC50 = 16000 nM T37848 CN93ZF 134138893 IC50 > 30000 nM T37848 C2A7CZ 134138904 IC50 = 12800 nM T37848 C78RUB 134138908 IC50 < 1000 nM T37848 CU8BV5 134139688 IC50 > 20000 nM T37848 CH3V9Q 134139925 IC50 > 25000 nM T37848 CTUZ02 134140953 IC50 = 7900 nM T37848 CQ2N5S 134141016 IC50 = 6900 nM T37848 C8TO1W 134142563 IC50 = 9300 nM T37848 C8MAB7 134142736 IC50 > 30000 nM T37848 CVC1Y4 134142943 IC50 = 12920 nM T37848 C2F9SA 134143025 IC50 = 11000 nM T37848 CU52XS 134143396 IC50 = 1500 nM T37848 CZ46SV 134145373 IC50 < 1000 nM T37848 CK13YN 134145788 IC50 > 30000 nM T37848 CS2DL8 134146184 EC50 = 2000 nM T37848 CF8CN2 134146399 IC50 = 8000 nM T37848 CWS36X 134147208 IC50 = 8400 nM T37848 CIST52 134147674 IC50 = 14000 nM T37848 C01DJX 134148367 IC50 = 5400 nM T37848 C0OHJ7 134148688 IC50 = 30000 nM T37848 CFG60Q 134148895 IC50 > 10000 nM T37848 CA5B2J 134150245 IC50 > 50000 nM T37848 C0S2VH 134150637 IC50 > 17000 nM T37848 C6NYU2 134150754 IC50 > 5000 nM T37848 COPA84 134151189 IC50 = 43000 nM T37848 C9NI7K 134151534 IC50 = 7700 nM T37848 CR2I8B 134151582 IC50 = 16000 nM T37848 CZH50T 134151855 IC50 > 30000 nM T37848 C8PT9W 134152052 IC50 > 30000 nM T37848 CGJ7B0 134152376 IC50 < 1000 nM T37848 C0N8OF 134152876 IC50 = 8700 nM T37848 CHWV04 134153381 IC50 < 1000 nM T37848 CP41RT 134154065 IC50 >= 20000 nM T37848 CM7X4P 134154315 IC50 = 23000 nM T37848 CB9F2G 134154510 IC50 = 15000 nM T37848 C0LGI2 134154676 IC50 > 30000 nM T37848 CZV9B3 134154775 IC50 > 30000 nM T37848 C0UEA6 134154910 IC50 = 9900 nM T37848 CA85UF 134155224 IC50 > 50000 nM T37848 CA49BH 134156727 IC50 > 50000 nM T37848 CJG0C4 134156793 IC50 = 5800 nM T37848 CM2BA7 134157196 IC50 = 30000 nM T37848 C7H8GQ 134157229 IC50 > 10000 nM T37848 C7AFS1 134157353 IC50 = 12000 nM T37848 CNS38M 134157776 IC50 = 21100 nM T37848 CK7B0U 134304087 IC50 > 10000 nM T37848 CX62UZ 134304119 IC50 > 10000 nM T37848 CUDY24 134304129 IC50 > 10000 nM T37848 CO5I4B 134304177 IC50 > 10000 nM T37848 CRD52S 134324842 IC50 > 10000 nM T37848 C17NBC 134325016 IC50 > 10000 nM T37848 CVLH60 134374993 IC50 = 300 nM T37848 C47TLY 134378796 IC50 = 12000 nM T37848 CFR87X 134477051 IC50 > 20000 nM T37848 CFYC29 134477061 IC50 = 20000 nM T37848 C20QBE 134477062 IC50 = 20000 nM T37848 CT58HM 134477070 IC50 = 430 nM T37848 C8W9YN 134477076 IC50 > 20000 nM T37848 CX5MS3 134477080 IC50 > 20000 nM T37848 CSO3Q9 134477081 IC50 > 20000 nM T37848 C32HVP 134477090 IC50 = 5900 nM T37848 CAED75 134477093 IC50 = 20000 nM T37848 CO15IT 134477094 IC50 = 20000 nM T37848 C0Q1MD 134477108 IC50 = 780 nM T37848 CX64SG 134477133 IC50 = 90 nM T37848 CT7J4U 134477136 IC50 = 20000 nM T37848 C51SKX 134477137 IC50 > 20000 nM T37848 CCVX65 134477139 IC50 > 20000 nM T37848 C03SFG 134477143 IC50 = 20000 nM T37848 C70XMC 134477147 IC50 = 20000 nM T37848 CL06KE 134477148 IC50 = 20000 nM T37848 C7JM1E 134477177 IC50 = 20000 nM T37848 C4LS2A 134477178 IC50 = 2300 nM T37848 CNU8M6 134477183 IC50 > 20000 nM T37848 CK9SR3 134477213 IC50 > 20000 nM T37848 C9WN3E 134477214 IC50 = 9000 nM T37848 C9IB8P 134477217 IC50 = 20000 nM T37848 CN37XZ 134477224 IC50 = 450 nM T37848 CR39TS 134477260 IC50 = 6700 nM T37848 CWNK85 134477261 IC50 = 6700 nM T37848 C9O5FS 134477264 IC50 > 20000 nM T37848 CS5ME8 134477268 IC50 > 20000 nM T37848 CC0OF9 134477275 IC50 > 20000 nM T37848 C1R9DV 134477283 IC50 = 270 nM T37848 CVR60G 134539903 IC50 > 25000 nM T37848 C20HAT 134585236 IC50 = 50000 nM T37848 C6W3VL 134585536 IC50 = 38000 nM T37848 CRL3O8 134585831 IC50 = 50000 nM T37848 CZB7I6 134821685 IC50 > 10000 nM T37848 CDC38O 134823958 IC50 = 80 nM T37848 CQI48P 135192983 IC50 = 20000 nM T37848 CT0GQ6 135197577 IC50 > 10000 nM T37848 C87VKA 135197594 IC50 > 10000 nM T37848 CQXS07 135197635 IC50 > 10000 nM T37848 C7KXF1 135197643 IC50 > 10000 nM T37848 CS4BM3 135236903 IC50 > 50000 nM T37848 CNEY95 135285657 IC50 > 50000 nM T37848 CA2OV3 135306913 IC50 > 50000 nM T37848 CH9RX5 135313574 IC50 = 58 nM T37848 CCJ97K 135313618 IC50 = 334 nM T37848 C76OJC 135313705 IC50 > 20000 nM T37848 C2L6PH 135313715 IC50 = 109 nM T37848 CO4W2L 135313730 IC50 > 20000 nM T37848 CQBZ60 135313773 IC50 = 4630 nM T37848 C3K2RL 135313899 IC50 = 200 nM T37848 CMR34P 135313919 IC50 = 12700 nM T37848 CR6K4Q 135313963 IC50 = 839 nM T37848 C9FNU5 135313965 IC50 = 9400 nM T37848 C75MZN 135314048 IC50 > 20000 nM T37848 CL12JU 135314107 IC50 = 1420 nM T37848 CPTO20 135314108 IC50 > 20000 nM T37848 C8Q4JP 135314141 IC50 > 20000 nM T37848 CXN1C7 135314251 IC50 = 1560 nM T37848 CBQ01J 135314252 IC50 = 1250 nM T37848 C9OZ3G 135314329 IC50 = 990 nM T37848 C46IBJ 135314337 IC50 = 442 nM T37848 CWI13E 135314362 IC50 > 20000 nM T37848 CI73PJ 135314386 IC50 = 59 nM T37848 CM3KV6 135314388 IC50 = 7440 nM T37848 CY24QI 135314390 IC50 = 350 nM T37848 CD64BJ 135314469 IC50 = 994 nM T37848 CW3DO8 135315463 IC50 > 50000 nM T37848 C75MTX 135315494 IC50 > 50000 nM T37848 CC49YE 135357669 IC50 = 26600 nM T37848 CS0UK5 135357843 IC50 = 47400 nM T37848 C76JPR 135405015 IC50 = 3000 nM T37848 C7K4PA 135412054 IC50 > 20000 nM T37848 C31VAN 135412231 IC50 > 20000 nM T37848 C47LAF 135418940 IC50 > 50000 nM T37848 CIS9K5 135421564 IC50 > 10000 nM T37848 CZJ62H 135423375 IC50 = 1100 nM T37848 CV8Q7A 135430397 IC50 = 5600 nM T37848 CZ4GP6 135446244 IC50 > 20000 nM T37848 CAJ2C0 135448904 IC50 = 2900 nM T37848 CA80OZ 135488014 IC50 = 4000 nM T37848 CDCF48 135488027 IC50 = 9000 nM T37848 CG5HY4 135507297 IC50 = 12000 nM T37848 C8QL5H 135508167 IC50 = 310 nM T37848 C3RX6B 135530418 IC50 = 80 nM T37848 CKF13W 135546072 IC50 > 10000 nM T37848 C65XMQ 135546228 IC50 = 6000 nM T37848 C8R4FB 135546884 IC50 > 20000 nM T37848 C7YA9M 135553232 IC50 = 3500 nM T37848 C15VPC 135553240 IC50 = 1400 nM T37848 CTB8U4 135553266 IC50 = 3700 nM T37848 CL9Q1F 135553267 IC50 = 11000 nM T37848 C6W3AL 135553268 IC50 = 1600 nM T37848 C53HFP 135553269 IC50 = 10000 nM T37848 C5Y6IB 135553271 IC50 = 2200 nM T37848 CY4MV6 135566354 IC50 > 50000 nM T37848 C24ZGX 135566644 IC50 > 40000 nM T37848 C2QDV5 135566741 IC50 = 40000 nM T37848 C8DX9H 135567148 IC50 = 11300 nM T37848 C23IWG 135567151 IC50 > 25000 nM T37848 CN1T7U 135681590 IC50 = 35000 nM T37848 CJ4C1Y 135681596 IC50 = 710 nM T37848 CJZ39U 135681612 IC50 < 46 nM T37848 C3EKM9 135681730 IC50 = 15000 nM T37848 C9UGN1 135681832 IC50 = 16000 nM T37848 C62NOS 135681833 IC50 = 4300 nM T37848 C3D0CJ 135681834 IC50 = 360 nM T37848 CIG3R9 135681875 IC50 = 13000 nM T37848 CCNH91 135743577 IC50 = 2610 nM T37848 CC9AU4 135869565 IC50 = 2100 nM T37848 CQSV28 135875708 IC50 = 14000 nM T37848 CF16XL 135875709 IC50 = 11000 nM T37848 CL35XZ 135875710 IC50 = 28000 nM T37848 C56WCS 135875711 IC50 = 7700 nM T37848 C37BGJ 135875712 IC50 = 10000 nM T37848 C9B5PC 135875713 IC50 = 40000 nM T37848 CACB27 135875714 IC50 = 23000 nM T37848 CKN2G0 135875715 IC50 = 19500 nM T37848 CCK5I3 135883253 IC50 > 10000 nM T37848 CU5VY1 135922386 IC50 = 4.1 nM T37848 C14OBQ 135928469 IC50 > 20000 nM T37848 C01HMT 135932346 IC50 = 2700 nM T37848 CBW3M8 135934887 IC50 = 1000 nM T37848 CA39ZG 135934888 IC50 = 700 nM T37848 CCIJ86 135960711 IC50 = 0.4 nM T37848 C6GS3B 135960712 IC50 = 1 nM T37848 CI9UP7 135960713 IC50 = 0.9 nM T37848 C4RY9Q 135960714 IC50 = 1.3 nM T37848 CWAH57 135960715 IC50 = 700 nM T37848 C36BQL 135960716 IC50 = 2.6 nM T37848 CVTF95 135960717 IC50 = 3.9 nM T37848 C01OML 135960718 IC50 = 4.5 nM T37848 C2G3JT 135960719 IC50 = 0.7 nM T37848 CI43OS 135960720 IC50 = 0.5 nM T37848 C6SZX2 135960721 IC50 = 1 nM T37848 C6E8WK 135960722 IC50 = 3.1 nM T37848 CZU46W 135960723 IC50 = 0.5 nM T37848 CUV5Q8 135960724 IC50 = 2.4 nM T37848 CFP18N 135960725 IC50 = 0.8 nM T37848 C4Z2CT 135960726 IC50 = 5.6 nM T37848 C3ST5C 135960727 IC50 = 3 nM T37848 CH4OX3 135960728 IC50 = 1.7 nM T37848 CVN7A3 135960729 IC50 = 3500 nM T37848 CQ8BM7 135960730 IC50 = 2.4 nM T37848 CA26EL 135960731 IC50 = 1.8 nM T37848 C9GUD2 135960732 IC50 = 19 nM T37848 C3KU5W 135960733 IC50 = 40 nM T37848 C4RL7Q 135985508 IC50 = 10000 nM T37848 C1ZT4N 135988927 IC50 = 800 nM T37848 C86BZJ 135988997 IC50 = 940 nM T37848 CEGJ60 136007966 IC50 = 6800 nM T37848 CKC95O 136036546 IC50 = 1900 nM T37848 CXH63V 136041747 IC50 > 40000 nM T37848 C6B5TC 136041748 IC50 > 40000 nM T37848 CU6XG1 136041749 IC50 > 40000 nM T37848 C74PRL 136041753 IC50 > 40000 nM T37848 CT4FJ1 136041757 IC50 = 40000 nM T37848 CEZP21 136041762 IC50 > 40000 nM T37848 CX67QW 136041765 IC50 > 40000 nM T37848 CM65BS 136041773 IC50 > 40000 nM T37848 C6P7JB 136041775 IC50 > 40000 nM T37848 C5CJF7 136041776 IC50 > 40000 nM T37848 CZ3BN1 136041792 IC50 = 40000 nM T37848 CG19DI 136041799 IC50 > 40000 nM T37848 CXJA29 136041804 IC50 = 40000 nM T37848 CHT31V 136041805 IC50 = 40000 nM T37848 CO8C4J 136041817 IC50 = 40000 nM T37848 C4QU6G 136041827 IC50 = 40000 nM T37848 CNE10X 136041834 IC50 = 40000 nM T37848 CS3AE1 136041847 IC50 = 40000 nM T37848 CZC47Y 136041848 IC50 = 40000 nM T37848 C4HJ7D 136044076 IC50 > 10000 nM T37848 C0RU6A 136053698 IC50 = 300 nM T37848 C83QVU 136056460 IC50 = 1200 nM T37848 CT57ZH 136069450 IC50 > 50000 nM T37848 CFT9R3 136069453 IC50 > 50000 nM T37848 CRPQ42 136069494 IC50 = 69000 nM T37848 CK8Z3V 136069521 IC50 = 40000 nM T37848 CPY1B2 136069522 IC50 > 50000 nM T37848 CX0OM4 136069523 IC50 > 50000 nM T37848 C6EU4D 136069524 IC50 > 50000 nM T37848 CQA2Z1 136069531 IC50 > 50000 nM T37848 CCH31A 136069532 IC50 > 50000 nM T37848 CQ1FS4 136069563 IC50 > 50000 nM T37848 CA91JG 136069599 IC50 = 40000 nM T37848 CGAB91 136069600 IC50 = 40000 nM T37848 C3ZAW2 136069605 IC50 = 40000 nM T37848 C8JXL5 136069609 IC50 = 31000 nM T37848 C9I0EQ 136069610 IC50 = 11000 nM T37848 C25EYJ 136069611 IC50 = 40000 nM T37848 CUE5X4 136086708 IC50 = 600 nM T37848 C80OJT 136086709 IC50 = 3300 nM T37848 CY79BE 136086710 IC50 = 1900 nM T37848 C2V8WH 136086711 IC50 = 2600 nM T37848 C1EAF5 136086712 IC50 = 2400 nM T37848 C5M6UO 136086713 IC50 = 450 nM T37848 CNEF50 136086718 IC50 = 2200 nM T37848 CE9A5G 136086719 IC50 = 1100 nM T37848 C27XOJ 136086720 IC50 = 800 nM T37848 C0K7PC 136086721 IC50 = 800 nM T37848 CC1DW7 136086722 IC50 = 1900 nM T37848 C14APV 136086723 IC50 = 700 nM T37848 C3N5RQ 136086724 IC50 = 1000 nM T37848 C69JHW 136117992 IC50 = 60 nM T37848 C63VTD 136118015 IC50 = 3100 nM T37848 CL08HS 136118016 IC50 = 6300 nM T37848 CTSB03 136118017 IC50 = 3600 nM T37848 CIR40T 136164062 IC50 = 3000 nM T37848 CD3F6B 136164063 IC50 = 2200 nM T37848 C4YK0X 136164064 IC50 = 18000 nM T37848 C19XOR 136164065 IC50 > 4400 nM T37848 CD0G5X 136164066 IC50 = 16000 nM T37848 C67AIH 136164067 IC50 > 13000 nM T37848 CBU8W6 136164068 IC50 = 500 nM T37848 C6LR7Y 136167037 IC50 > 50000 nM T37848 CGX6C4 136173253 IC50 > 100000 nM T37848 CC4UM3 136176116 IC50 > 40000 nM T37848 CJRK81 136176117 IC50 > 40000 nM T37848 C63IOS 136176118 IC50 > 40000 nM T37848 CP2YM7 136176127 IC50 > 40000 nM T37848 C8XIJ0 136176128 IC50 = 19000 nM T37848 C4WG2F 136176132 IC50 > 40000 nM T37848 C1LK9U 136183381 IC50 = 40000 nM T37848 CC52HL 136189674 IC50 > 20000 nM T37848 CQTB32 136205798 IC50 > 10000 nM T37848 CV8QP3 136205832 IC50 > 50000 nM T37848 CB93EM 136205833 IC50 > 50000 nM T37848 CDEX74 136229147 IC50 = 700 nM T37848 CRET01 136230229 IC50 = 40000 nM T37848 CX1KI8 136230230 IC50 = 40000 nM T37848 CUE6N8 136230232 IC50 = 40000 nM T37848 C8Q1AP 136230233 IC50 = 40000 nM T37848 C70RXE 136230234 IC50 = 40000 nM T37848 C4W0KN 136230235 IC50 = 40000 nM T37848 CBS97C 136239447 IC50 = 16000 nM T37848 CQ10OF 136240980 IC50 > 20000 nM T37848 CL4MO3 136249382 IC50 = 40000 nM T37848 C1HI5T 136264454 IC50 = 40000 nM T37848 CC8Q2D 136375233 IC50 = 10000 nM T37848 C4OVP2 136416802 IC50 > 50000 nM T37848 C7ZCT8 136416815 IC50 > 50000 nM T37848 C95TJH 136632047 IC50 > 10000 nM T37848 CI94YQ 136982007 IC50 > 10000 nM T37848 CK4CM2 137028369 IC50 > 50000 nM T37848 C7TAZ5 137142885 IC50 > 10000 nM T37848 C0UP1A 137174951 IC50 = 300 nM T37848 CO6WA9 137313834 IC50 > 50000 nM T37848 CE1G4P 137333984 IC50 = 7000 nM T37848 C0PL4B 137434175 IC50 > 30000 nM T37848 C8F4WH 137462364 EC50 > 20000 nM T37848 CO72JI 137521054 IC50 > 20000 nM T37848 CDLB52 137521232 IC50 > 20000 nM T37848 CP86HV 137521251 IC50 > 20000 nM T37848 CS34IR 137628304 IC50 = 10000 nM T37848 C9ACX4 137628305 IC50 < 10000 nM T37848 CP2C1J 137628306 IC50 > 25000 nM T37848 CDGB50 137628309 IC50 < 10000 nM T37848 CW8ZR6 137628310 IC50 < 10000 nM T37848 C48QKY 137628311 IC50 < 10000 nM T37848 CH5AV6 137628312 IC50 < 10000 nM T37848 CU9O3A 137628639 IC50 > 20000 nM T37848 CEZT29 137628641 IC50 > 10000 nM T37848 C6B5US 137628648 IC50 > 10000 nM T37848 C3A6PQ 137628670 IC50 > 10000 nM T37848 C6JO4G 137631841 IC50 > 20000 nM T37848 CH67OI 137631881 IC50 < 10000 nM T37848 C2XI8Y 137632393 IC50 = 280 nM T37848 CES7L0 137632608 IC50 > 20000 nM T37848 C6MRU3 137633431 IC50 > 20000 nM T37848 CV8M3P 137633531 IC50 = 17700 nM T37848 CN2BK8 137633559 IC50 = 10 nM T37848 CG91VC 137633656 IC50 = 685 nM T37848 C8C0OE 137634027 IC50 > 100000 nM T37848 CNU3O7 137634107 IC50 > 20000 nM T37848 COD07I 137634464 IC50 = 12900 nM T37848 C5PTM8 137634588 IC50 = 137800 nM T37848 CE9O8V 137634616 IC50 = 30000 nM T37848 CT8E0M 137635041 IC50 = 11300 nM T37848 CP07AG 137635043 IC50 = 11000 nM T37848 C8TU2S 137635295 IC50 = 36200 nM T37848 CA3WP9 137635668 IC50 = 440 nM T37848 C4ALG0 137635843 IC50 = 8561 nM T37848 CYL39G 137635979 IC50 > 10000 nM T37848 CBCQ18 137636228 IC50 = 60000 nM T37848 C6Y8VD 137636260 IC50 = 6526 nM T37848 CM51CG 137636524 IC50 = 4900 nM T37848 CH2SR6 137636922 IC50 = 5282 nM T37848 C52XYJ 137637143 IC50 > 200000 nM T37848 C5YV3A 137637566 IC50 = 20000 nM T37848 CH3M0S 137637752 IC50 = 6300 nM T37848 CR9IZ6 137637770 IC50 > 50000 nM T37848 CDBT63 137637838 IC50 = 6150 nM T37848 CFK9D8 137638117 IC50 = 6300 nM T37848 C21YPG 137638242 IC50 = 8450 nM T37848 CHGE26 137638325 IC50 = 74 nM T37848 C2Y9HF 137638913 IC50 > 20000 nM T37848 C0ZS9N 137638993 IC50 > 20000 nM T37848 C8WO2G 137639251 IC50 > 20000 nM T37848 CZ2A5K 137639461 IC50 = 17000 nM T37848 CF5TI6 137639661 IC50 = 27400 nM T37848 CYPQ38 137640446 IC50 > 20000 nM T37848 CV85YQ 137640474 IC50 > 20000 nM T37848 CKL78U 137640727 IC50 = 1710 nM T37848 CN1RV9 137640762 IC50 = 16500 nM T37848 C0Q4IM 137641652 IC50 > 20000 nM T37848 CYW61U 137641749 IC50 = 9290 nM T37848 CUJ08S 137642106 IC50 = 179 nM T37848 CH21YK 137642640 IC50 > 50000 nM T37848 CR9C5G 137642830 IC50 <= 20000 nM T37848 CO8V4W 137642907 IC50 > 20000 nM T37848 CUB38E 137642944 IC50 > 50000 nM T37848 CGA2S0 137643017 IC50 = 3 nM T37848 CJT81N 137643054 IC50 > 20000 nM T37848 CPW7T0 137643121 IC50 = 40100 nM T37848 C58ISN 137643139 IC50 = 10000 nM T37848 C1FU3P 137643308 IC50 > 20000 nM T37848 CVC3S2 137643317 IC50 > 20000 nM T37848 CHOI53 137643582 IC50 > 30000 nM T37848 CI2F1B 137644335 IC50 = 6010 nM T37848 CU91LQ 137644813 IC50 = 7830 nM T37848 CN97GA 137645181 IC50 > 10000 nM T37848 C1EKA8 137645415 IC50 = 94600 nM T37848 CNB72K 137645644 IC50 = 5500 nM T37848 CKT2R4 137646125 IC50 = 2780 nM T37848 CU47YW 137646415 IC50 > 20000 nM T37848 C5IHS8 137646440 IC50 > 20000 nM T37848 CN4U1A 137646732 IC50 > 30000 nM T37848 CDCH19 137646766 IC50 > 20000 nM T37848 CFKR53 137646837 IC50 = 20000 nM T37848 CRA48Q 137647184 IC50 = 2240 nM T37848 CLT73G 137647199 IC50 = 1500 nM T37848 CXS2U7 137647336 IC50 = 15200 nM T37848 CE57QM 137647529 IC50 > 20000 nM T37848 C42DRJ 137647643 IC50 = 1290 nM T37848 CLAR76 137647645 IC50 > 20000 nM T37848 CGW71J 137647660 IC50 > 50000 nM T37848 CUDM82 137647787 IC50 = 7100 nM T37848 C4AKD7 137647838 IC50 > 20000 nM T37848 C2SG0J 137648286 IC50 = 144 nM T37848 CP32AR 137648836 IC50 > 20000 nM T37848 CV03IF 137648903 IC50 < 10000 nM T37848 C5AT7D 137649062 IC50 > 20000 nM T37848 C3GP4Y 137649582 IC50 > 40000 nM T37848 C04JSE 137649716 IC50 > 50000 nM T37848 C8N9CH 137650363 IC50 = 37500 nM T37848 CL7ZX9 137651411 IC50 > 50000 nM T37848 CD9ZN4 137651429 IC50 > 20000 nM T37848 C2XNL7 137651646 IC50 = 8230 nM T37848 C6GJA5 137651722 IC50 > 53000 nM T37848 C2JBS1 137651899 IC50 > 100000 nM T37848 C2L7ZT 137652982 IC50 = 4500 nM T37848 CKV03G 137653074 IC50 > 30000 nM T37848 CK14LN 137653163 IC50 = 7900 nM T37848 C38FXZ 137653443 IC50 > 20000 nM T37848 C6MJU7 137653906 IC50 = 9032 nM T37848 CV59RY 137654290 IC50 = 5580 nM T37848 C9TQ5P 137654575 IC50 = 15 nM T37848 CHB2F0 137654670 IC50 = 11900 nM T37848 CMXL93 137655135 IC50 = 1400 nM T37848 CX5YF2 137655402 IC50 = 1400 nM T37848 CSRK73 137655508 IC50 = 46000 nM T37848 C17LIA 137655641 IC50 > 33000 nM T37848 CJ7D8K 137655914 IC50 > 20000 nM T37848 C0N6KU 137655916 IC50 = 6309.57 nM T37848 CRY40J 137655938 IC50 = 12700 nM T37848 C1OXG8 137655944 IC50 > 10000 nM T37848 CZ4W3T 137656391 IC50 > 50000 nM T37848 C29UVL 137656780 IC50 = 10800 nM T37848 C8DT1W 137657247 IC50 > 20000 nM T37848 CU28CY 137657424 IC50 > 20000 nM T37848 C2BGF3 137657547 IC50 = 622 nM T37848 CB61UY 137658460 IC50 > 20000 nM T37848 CG96FH 137658637 IC50 > 10000 nM T37848 CL45EH 137658689 IC50 = 7897 nM T37848 CURX53 137658725 IC50 = 70 nM T37848 C1R7UP 137658901 IC50 = 19200 nM T37848 CKVH89 137658916 IC50 = 2200 nM T37848 CJ8L1W 137659170 IC50 > 50000 nM T37848 CH4M3X 137659806 IC50 = 13700 nM T37848 CS38RA 137660718 IC50 = 155700 nM T37848 CA4MT5 137661210 IC50 = 1850 nM T37848 C0XCS4 137661956 IC50 = 3600 nM T37848 C96QPV 137662004 IC50 > 5000 nM T37848 CSEZ59 137662026 IC50 = 11700 nM T37848 C6KYD7 137700754 IC50 > 10000 nM T37848 C9MNG4 138319677 IC50 > 10000 nM T37848 CJC95O 138319684 IC50 > 50000 nM T37848 CPTE92 138319693 IC50 > 10000 nM T37848 CMP8U3 138376515 IC50 > 10000 nM T37848 CE79SV 138377584 IC50 > 50000 nM T37848 CB8FE3 138393376 IC50 > 5000 nM T37848 CKDZ26 138504497 IC50 > 30000 nM T37848 C1XSH7 138594194 IC50 > 10000 nM T37848 CG4RO6 138632227 IC50 > 18000 nM T37848 CHT39X 138632268 IC50 > 18000 nM T37848 CVB6L2 138632650 IC50 > 18000 nM T37848 CN9R4A 138691364 IC50 = 310 nM T37848 CI9YB7 138753112 IC50 = 3030 nM T37848 C7EKA2 138911324 IC50 > 10000 nM T37848 C1BOT2 139030270 IC50 = 8900 nM T37848 CAF2H8 139488606 IC50 = 100 nM T37848 CD29IP 139507088 IC50 > 10000 nM T37848 CF8LN1 139582020 IC50 > 30000 nM T37848 CI1D9F 139600335 IC50 > 100000 nM T37848 CG2NH6 139600336 IC50 > 20000 nM T37848 C0HN5J 139600337 IC50 > 20000 nM T37848 CGA12N 141473855 IC50 = 37690 nM T37848 C2YC6F 141473885 IC50 = 36880 nM T37848 C9JSZ2 141529337 IC50 > 10000 nM T37848 CSE1D2 141529338 IC50 > 10000 nM T37848 C43LDR 141730928 IC50 > 50000 nM T37848 C2D9TE 141756938 IC50 = 4000 nM T37848 C53UZY 141757055 IC50 = 100 nM T37848 C06ZBJ 142416740 IC50 > 20000 nM T37848 C9J1ZO 142416754 IC50 = 12000 nM T37848 C58KQF 142416884 IC50 > 20000 nM T37848 C68OXK 142416914 IC50 = 1800 nM T37848 C7C3MK 142416935 IC50 > 20000 nM T37848 CO7DK2 142416967 IC50 = 10000 nM T37848 C17XZS 142727681 IC50 = 3520 nM T37848 C1UCX0 144953608 IC50 > 10000 nM T37848 C9GRB2 144953612 IC50 > 10000 nM T37848 CV4X5P 144953614 IC50 > 10000 nM T37848 C1W8QR 145865307 IC50 > 50000 nM T37848 C6VB3O 145925651 IC50 > 50118.72 nM T37848 C9ISH6 145925685 IC50 > 20000 nM T37848 CL8VT0 145946399 IC50 > 20000 nM T37848 CVND41 145949156 IC50 > 20000 nM T37848 CF1MH2 145949267 IC50 > 30000 nM T37848 CI14LP 145949343 IC50 > 12000 nM T37848 CXJ07F 145949470 IC50 > 25000 nM T37848 C8KA6P 145949486 IC50 > 20000 nM T37848 CA0B3D 145949907 IC50 > 20000 nM T37848 C7W9ZT 145949949 IC50 > 20000 nM T37848 CI3V6Y 145950358 IC50 = 5600 nM T37848 COG04E 145950432 IC50 = 13000 nM T37848 CAWU95 145950510 IC50 > 20000 nM T37848 CLZ54T 145950740 IC50 > 50000 nM T37848 CL2OR1 145950976 IC50 > 20000 nM T37848 C4FM3C 145951105 IC50 > 50000 nM T37848 CLV0G6 145951167 IC50 = 29000 nM T37848 C2M8PI 145951236 IC50 > 20000 nM T37848 CH0K8V 145951521 IC50 = 6800 nM T37848 C3OMF2 145951963 IC50 = 2400 nM T37848 CG5OW3 145951998 IC50 = 92000 nM T37848 CEB71V 145952023 IC50 > 30000 nM T37848 C4LJV9 145952024 IC50 = 214000 nM T37848 C1QA6W 145952070 IC50 = 181000 nM T37848 CC7IP8 145952109 IC50 = 6400 nM T37848 CN0S3B 145952357 IC50 = 24000 nM T37848 C3E5BK 145952508 IC50 > 10000 nM T37848 CC4K9F 145952601 IC50 > 20000 nM T37848 C0RGQ7 145952699 IC50 > 10000 nM T37848 CGW92C 145952721 IC50 > 12000 nM T37848 C2FXL5 145952723 IC50 = 3350 nM T37848 C9D5MZ 145952745 IC50 > 50000 nM T37848 CRN85T 145952991 IC50 > 25000 nM T37848 CER83S 145953040 IC50 > 20000 nM T37848 CA7W2O 145953059 IC50 = 4900 nM T37848 C1A4CH 145953177 IC50 = 4230 nM T37848 COZ1F4 145953325 IC50 > 20000 nM T37848 C09WNF 145953342 IC50 > 12000 nM T37848 CEJ26X 145953403 IC50 > 20000 nM T37848 CS21ZB 145953739 IC50 > 20000 nM T37848 C5LB7M 145953999 IC50 = 90000 nM T37848 CW9I0R 145954143 IC50 > 10000 nM T37848 CPW52X 145954567 IC50 = 11000 nM T37848 CN5L4K 145954640 IC50 = 24000 nM T37848 C59AVT 145954818 IC50 > 20000 nM T37848 C4P6MT 145954878 IC50 = 3160 nM T37848 CWA8H2 145955288 IC50 > 30000 nM T37848 CQ5SN1 145955289 IC50 = 7000 nM T37848 CK0S1G 145955694 IC50 > 20000 nM T37848 CE03RK 145955745 IC50 = 5620 nM T37848 CF6T7G 145955884 IC50 > 20000 nM T37848 C0HN4S 145955917 IC50 = 12000 nM T37848 C8RYI4 145956153 IC50 > 10000 nM T37848 C8Y4VT 145956312 IC50 > 20000 nM T37848 C4G6XJ 145956824 IC50 > 20000 nM T37848 C7N6CA 145956935 IC50 = 5200 nM T37848 CBFU43 145957229 IC50 = 13000 nM T37848 CQ0JP4 145957239 IC50 > 20000 nM T37848 CK94HO 145957365 IC50 > 12000 nM T37848 CE1G7A 145957474 IC50 = 17243 nM T37848 C70LMY 145957553 IC50 > 20000 nM T37848 C20EDK 145957568 IC50 = 42000 nM T37848 CFZJ34 145957574 IC50 > 19952.62 nM T37848 CB2K0W 145957599 IC50 = 6790 nM T37848 C3B0YE 145957778 IC50 = 11000 nM T37848 CID3G5 145958087 IC50 > 50000 nM T37848 C8WZY3 145958093 IC50 > 12000 nM T37848 CXHM49 145958111 IC50 > 20000 nM T37848 CBC1T9 145958296 IC50 > 20000 nM T37848 C3TX8O 145958528 IC50 > 12000 nM T37848 CM8U9A 145958674 IC50 = 29000 nM T37848 CT3U1A 145958698 IC50 = 2210 nM T37848 CBF54O 145958967 IC50 > 25000 nM T37848 CB5XW7 145959080 IC50 = 5200 nM T37848 CH47WN 145959135 IC50 = 19000 nM T37848 CW8M0I 145959142 IC50 > 20000 nM T37848 CLS3W5 145959177 IC50 > 25000 nM T37848 C8DH5F 145959814 IC50 > 12000 nM T37848 C5Z9US 145959844 IC50 > 20000 nM T37848 CLJE41 145959897 IC50 > 25000 nM T37848 CW1GO5 145960043 IC50 = 39000 nM T37848 CUD9E6 145960079 IC50 > 20000 nM T37848 CI8Q2V 145960175 IC50 = 15000 nM T37848 C3F8XM 145960247 IC50 > 20000 nM T37848 CDKY72 145960338 IC50 = 39000 nM T37848 CT6OH1 145960389 IC50 = 8380 nM T37848 C0WB6J 145960881 IC50 > 20000 nM T37848 C5ZD1H 145961500 IC50 > 30000 nM T37848 CD01PX 145961863 IC50 > 20000 nM T37848 C42PLT 145962320 IC50 = 45500 nM T37848 CDY47R 145962388 IC50 = 5810 nM T37848 CQ2TN4 145962919 IC50 > 30000 nM T37848 CKLA91 145962920 IC50 = 4300 nM T37848 C64OLM 145963140 IC50 > 20000 nM T37848 CU8Y2C 145963537 IC50 > 20000 nM T37848 C62MVS 145964029 IC50 > 50000 nM T37848 CFC8Q4 145964097 IC50 > 10000 nM T37848 CFAK41 145964101 IC50 = 50000 nM T37848 C2IM3V 145964416 IC50 > 10000 nM T37848 CQ5XM3 145964429 IC50 > 10000 nM T37848 CTJI01 145964752 IC50 > 20000 nM T37848 CQA98S 145964789 IC50 = 140 nM T37848 CRZ5T1 145964880 IC50 > 10000 nM T37848 CQZ3F7 145965198 IC50 > 20000 nM T37848 CSK8Y1 145965486 IC50 = 33000 nM T37848 C4P7UD 145965756 IC50 = 16500 nM T37848 C42FZC 145966011 IC50 > 20000 nM T37848 C2MS3R 145966170 IC50 >= 30000 nM T37848 CZ9AG8 145966405 IC50 = 7760 nM T37848 CRS65V 145966585 IC50 > 10000 nM T37848 C4V5QG 145966727 IC50 = 10000 nM T37848 CPH9E3 145967023 IC50 = 3600 nM T37848 CW02FZ 145967133 IC50 > 10000 nM T37848 C3K7QC 145967522 IC50 > 10000 nM T37848 CC0QA2 145967606 IC50 > 20000 nM T37848 CTGF42 145967808 IC50 > 10000 nM T37848 C19IVD 145967885 IC50 = 17000 nM T37848 CR36FU 145968121 IC50 = 6900 nM T37848 CNB7G5 145968344 IC50 = 9700 nM T37848 CX42BV 145968371 IC50 = 7270 nM T37848 CQCY49 145968539 IC50 > 10000 nM T37848 C7MAX3 145968702 IC50 > 30000 nM T37848 CQJP12 145968722 IC50 = 300 nM T37848 CU6RH3 145968879 IC50 = 14600 nM T37848 CJUK65 145968931 IC50 > 10000 nM T37848 CCB21N 145969176 IC50 = 8500 nM T37848 CNH7O5 145969326 IC50 = 158.49 nM T37848 C4HF5M 145969366 IC50 = 5100 nM T37848 CUI97C 145969471 IC50 > 10000 nM T37848 C6TDW9 145969499 IC50 > 10000 nM T37848 C9TWE2 145969541 IC50 > 10000 nM T37848 C94URS 145969597 IC50 > 50000 nM T37848 CHZ7N3 145969706 IC50 = 630.96 nM T37848 C2S8DE 145969909 IC50 > 20000 nM T37848 C59ZFQ 145970027 IC50 > 10000 nM T37848 C0WIZ5 145970221 IC50 > 10000 nM T37848 CI3O2K 145970611 IC50 > 20000 nM T37848 C8B4IY 145970709 IC50 > 10000 nM T37848 C6CD4Z 145970793 IC50 > 20000 nM T37848 CS5U3M 145970807 IC50 > 20000 nM T37848 C5O2EA 145971149 IC50 > 10000 nM T37848 CND2K7 145971189 IC50 > 20000 nM T37848 CMI45E 145971507 IC50 > 20000 nM T37848 CXF9E7 145972420 IC50 = 5300 nM T37848 CU13IP 145972573 IC50 > 10000 nM T37848 CP7LW2 145973146 IC50 = 1780 nM T37848 CV9OM2 145973260 IC50 > 10000 nM T37848 C8RFM3 145973261 IC50 > 20000 nM T37848 C8OSM0 145973345 IC50 > 20000 nM T37848 C6OI3K 145973962 IC50 > 10000 nM T37848 C4XZ1W 145973987 IC50 = 21600 nM T37848 C56HYE 145974067 IC50 = 37000 nM T37848 C54QHK 145974080 IC50 > 20000 nM T37848 CH5CL0 145974084 IC50 > 10000 nM T37848 CJN96Q 145974556 IC50 = 39000 nM T37848 C0Q2NJ 145974673 IC50 = 440 nM T37848 C80VHP 145974690 IC50 > 10000 nM T37848 CGWM29 145974840 IC50 = 50000 nM T37848 C9G2OD 145974857 IC50 = 8570 nM T37848 CAU82Y 145975252 IC50 > 10000 nM T37848 CSBQ67 145975261 IC50 > 10000 nM T37848 C2B4EW 145975334 IC50 = 1279 nM T37848 CPM02H 145975616 IC50 = 1600 nM T37848 CUZ47S 145975654 IC50 = 6700 nM T37848 CQ2H6F 145976125 IC50 > 10000 nM T37848 C9MK4Z 145976157 IC50 = 10000 nM T37848 C4RO6S 145976616 IC50 > 50000 nM T37848 C5R7ZH 145977058 IC50 > 10000 nM T37848 C0IQV7 145977447 IC50 = 49 nM T37848 CUV49K 145977796 IC50 = 43400 nM T37848 CWJ46S 145978007 IC50 > 20000 nM T37848 CAS46P 145978366 IC50 = 4600 nM T37848 C4XV7J 145978553 IC50 = 9900 nM T37848 C3S0UI 145978581 IC50 = 50000 nM T37848 C01PMA 145979438 IC50 = 1200 nM T37848 C2D5YT 145980015 IC50 = 1200 nM T37848 CWA6L3 145981037 IC50 > 20000 nM T37848 CB7LD6 145981185 IC50 = 900 nM T37848 CGA83C 145981271 IC50 > 10000 nM T37848 C79EQW 145981356 IC50 = 900 nM T37848 CA0Y1X 145981628 IC50 = 1600 nM T37848 CLG9V4 145982062 IC50 > 30000 nM T37848 CAJQ81 145983214 IC50 = 6400 nM T37848 CJ35DM 145984299 IC50 = 23000 nM T37848 C4HAP0 145984727 IC50 = 12300 nM T37848 CTL5Y0 145986900 IC50 = 1000 nM T37848 COB69L 145987073 IC50 = 600 nM T37848 C5R6BS 145987142 IC50 > 10000 nM T37848 C78MWI 145987354 IC50 = 230 nM T37848 C7O1PF 145987480 IC50 > 20000 nM T37848 C81LEH 145987485 IC50 > 20000 nM T37848 CMRQ02 145987862 IC50 > 20000 nM T37848 CUAY25 145988620 IC50 > 10000 nM T37848 CY3MR0 145989049 IC50 > 10000 nM T37848 CHTG87 145989489 IC50 = 7800 nM T37848 C70HDR 145989886 IC50 = 11000 nM T37848 C8RGA4 145990244 IC50 = 5700 nM T37848 C7GK3H 145990715 IC50 > 100000 nM T37848 C0KNI4 145991888 IC50 = 1600 nM T37848 CE1L5T 145992719 IC50 > 20000 nM T37848 C3PD7L 145992760 IC50 = 13000 nM T37848 CA1QE7 145993306 IC50 > 30000 nM T37848 CMIH10 145993513 IC50 > 20000 nM T37848 CH3EP0 145993573 IC50 = 5500 nM T37848 CY37RJ 145994215 IC50 = 700 nM T37848 CHJ79V 145997874 IC50 > 10000 nM T37848 CAU3Z1 146020618 IC50 = 19700 nM T37848 C7F6SU 146047134 IC50 > 200000 nM T37848 CBRE71 146047136 IC50 > 20000 nM T37848 C2RJ1U 146176418 IC50 > 50000 nM T37848 C5VOC0 146431408 IC50 = 1022.3 nM T37848 CS54CM 146433251 IC50 > 40000 nM T37848 CGO5C4 146433253 IC50 > 40000 nM T37848 C61LGO 146433463 IC50 = 4200 nM T37848 C4OSN5 146433538 IC50 > 40000 nM T37848 CN2MA4 146433574 IC50 = 4200 nM T37848 C5ZOJ3 146680920 IC50 = 26000 nM T37848 C9YJZ5 147180858 IC50 = 7950 nM T37848 CUAY08 148018738 IC50 > 10000 nM T37848 CQK39B 149491764 IC50 > 10000 nM T37848 C1ZX5D 149494192 IC50 > 10000 nM T37848 CL6T4P 149986651 IC50 = 1400 nM T37848 CTI5R1 151961601 IC50 = 6470 nM T37848 CC3ME1 152131905 IC50 < 1000 nM T37848 C36ISR 153434865 IC50 > 10000 nM T37848 CG5IF7 154701259 IC50 > 1000 nM T37848 CZE1S5 155126870 IC50 > 50000 nM T37848 CI6EB5 155126882 IC50 > 50000 nM T37848 CF2CU8 155510758 IC50 > 30000 nM T37848 CG5HO8 155511239 IC50 > 100000 nM T37848 C7ZE5Q 155511547 IC50 = 2000 nM T37848 C1WRE2 155511764 IC50 > 100000 nM T37848 CQ83KZ 155512662 IC50 > 10000 nM T37848 CSL73Z 155513136 IC50 > 794.33 nM T37848 C5M6NS 155513226 IC50 > 27000 nM T37848 C8SW9I 155513332 IC50 = 900 nM T37848 C17RIB 155513592 IC50 > 20000 nM T37848 CT74QE 155513632 IC50 = 2000 nM T37848 CPU81W 155513803 IC50 > 25000 nM T37848 CPE58H 155514125 IC50 > 20000 nM T37848 CZUP45 155514353 IC50 > 30000 nM T37848 CL41JO 155514699 IC50 > 25000 nM T37848 CD53LC 155514863 IC50 > 25000 nM T37848 C9HG0U 155515457 IC50 > 20000 nM T37848 CMZ4Q7 155515478 IC50 > 25000 nM T37848 CYD75Z 155515691 IC50 = 351.2 nM T37848 CDP7E5 155516065 IC50 = 6309.57 nM T37848 C7OF4C 155516118 IC50 = 7800 nM T37848 CCJ14L 155516448 IC50 = 210 nM T37848 CPUG37 155516479 IC50 > 50000 nM T37848 C49INQ 155516757 IC50 = 4050 nM T37848 CY0CK6 155516843 IC50 > 50118.72 nM T37848 CL9IN5 155516936 IC50 > 25000 nM T37848 CA3K9P 155517032 IC50 < 10000 nM T37848 C0KI2X 155517513 IC50 = 2000 nM T37848 CQ52LM 155518361 IC50 = 5400 nM T37848 CRD79Z 155518589 IC50 = 10000 nM T37848 CAL54I 155518651 IC50 = 1258.93 nM T37848 C30SPO 155518654 IC50 = 49000 nM T37848 CVH0P8 155519454 IC50 = 10000 nM T37848 C0KLD8 155519559 IC50 = 20000 nM T37848 C1U3CL 155520250 IC50 = 12900 nM T37848 C8LP0E 155520285 IC50 = 3110 nM T37848 CF19DM 155521087 IC50 > 30000 nM T37848 CI9U3X 155521508 IC50 = 16000 nM T37848 CK7RM1 155521671 IC50 = 5200 nM T37848 C8J9GQ 155521846 IC50 > 25000 nM T37848 C0ZXV4 155522886 IC50 = 10000 nM T37848 C5N0GE 155523029 IC50 > 50118.72 nM T37848 CC5GO1 155523088 IC50 = 7820 nM T37848 C2LO4Y 155523731 IC50 < 10000 nM T37848 C3LC2H 155523754 IC50 > 20000 nM T37848 C12KNB 155523817 IC50 = 80 nM T37848 CYI71L 155523951 IC50 = 35500 nM T37848 CGK3T7 155524130 IC50 = 8400 nM T37848 CTU67Z 155524559 IC50 > 100000 nM T37848 CFM45O 155524794 IC50 = 2300 nM T37848 C3T4EL 155524825 IC50 = 4800 nM T37848 CN9QW1 155525049 IC50 > 25000 nM T37848 CG71WI 155525128 IC50 < 10000 nM T37848 C6J3DF 155525653 IC50 > 25000 nM T37848 CZW45D 155525803 IC50 = 6309.57 nM T37848 CA34FW 155526470 IC50 = 5140 nM T37848 CI31SP 155527821 IC50 = 19600 nM T37848 C05QTC 155528035 IC50 = 10000 nM T37848 C0B2NV 155528644 IC50 = 13000 nM T37848 CVW07K 155528897 IC50 > 100000 nM T37848 C5QA2B 155529241 IC50 < 10000 nM T37848 C9U8FN 155529326 IC50 = 18400 nM T37848 CW5TM8 155529670 IC50 = 19952.62 nM T37848 C7SEX2 155529894 IC50 = 4700 nM T37848 C4F7WU 155530183 IC50 = 27840 nM T37848 CK5X2E 155530190 IC50 > 20000 nM T37848 CQ6F7O 155530369 IC50 < 10000 nM T37848 CQD26H 155530468 IC50 > 20000 nM T37848 C1HFK3 155530973 IC50 >= 2500 nM T37848 CZG2O7 155532057 IC50 = 14900 nM T37848 C3U6VQ 155532120 IC50 > 50118.72 nM T37848 CH62TN 155532900 IC50 = 1400 nM T37848 C4V5SB 155533390 IC50 > 50118.72 nM T37848 C3DR2V 155533849 IC50 = 4690 nM T37848 C2QB7A 155534427 IC50 = 3981.07 nM T37848 CPXV81 155534530 IC50 = 127.2 nM T37848 CR6VT8 155534625 IC50 = 3162.28 nM T37848 C63HSA 155534748 IC50 > 50000 nM T37848 CIF97P 155535006 IC50 > 50118.72 nM T37848 C6QV5A 155535350 IC50 >= 2500 nM T37848 CX7PM4 155535638 IC50 = 3981.07 nM T37848 CTH8B9 155535743 IC50 > 20000 nM T37848 C9FPB6 155535794 IC50 = 8700 nM T37848 CY97DN 155535886 IC50 = 12800 nM T37848 C7FVE8 155537034 IC50 = 3530 nM T37848 CQU0H3 155537238 IC50 = 1000 nM T37848 CM1BX0 155537411 IC50 = 4200 nM T37848 CC7B3P 155537582 IC50 = 2500 nM T37848 C8K3XJ 155537606 IC50 = 11900 nM T37848 CM3PB2 155537682 IC50 = 10000 nM T37848 CCO96S 155538113 IC50 > 100000 nM T37848 CDU52V 155538567 IC50 = 80 nM T37848 CUS3I9 155538644 IC50 < 10000 nM T37848 CY8MZ6 155538967 IC50 = 3981.07 nM T37848 C1FZY9 155539610 IC50 = 42.9 nM T37848 C41LEI 155539901 IC50 > 10000 nM T37848 CW0XH5 155539949 IC50 > 10000 nM T37848 C9HOF6 155540194 IC50 = 1584.89 nM T37848 CGH8T5 155540333 IC50 > 10000 nM T37848 CB43YR 155540395 IC50 > 40000 nM T37848 CDQF20 155540443 IC50 > 30000 nM T37848 CW2V3F 155540455 IC50 = 1600 nM T37848 C0OGZ2 155540539 IC50 = 15848.93 nM T37848 C9YO0E 155540667 IC50 = 3040 nM T37848 CE74PT 155541294 IC50 = 332 nM T37848 CP2K9D 155541549 IC50 > 10000 nM T37848 CL18DI 155542104 IC50 > 10000 nM T37848 C5T9KE 155542416 IC50 > 50000 nM T37848 CIPG54 155542639 IC50 > 10000 nM T37848 C1SY0G 155543154 IC50 > 27000 nM T37848 CNY60D 155543679 IC50 > 10000 nM T37848 CNH46F 155543687 IC50 > 40000 nM T37848 C4M6YT 155544005 IC50 = 1995.26 nM T37848 C1S6GK 155546762 IC50 > 25000 nM T37848 CH94MI 155547266 IC50 > 10000 nM T37848 CQ6D2C 155547369 IC50 > 25000 nM T37848 CQ62MW 155547536 IC50 > 10000 nM T37848 C7GSO4 155548469 IC50 = 7320 nM T37848 CRY3A2 155548898 IC50 > 30000 nM T37848 CH25ZD 155549064 IC50 > 50000 nM T37848 CJD38X 155549583 IC50 = 10000 nM T37848 C08YOZ 155549638 IC50 = 3700 nM T37848 CS83IV 155550025 IC50 > 25000 nM T37848 CD4PW8 155550069 IC50 = 9700 nM T37848 C8NQ0I 155550263 IC50 < 1584.89 nM T37848 CHDG36 155550819 IC50 > 25000 nM T37848 C6JV3E 155551216 IC50 = 3300 nM T37848 C2K1OB 155551593 IC50 > 25000 nM T37848 CGDS14 155551776 IC50 > 20000 nM T37848 C2UYP0 155552120 IC50 = 1312.3 nM T37848 CEN80B 155552714 IC50 > 10000 nM T37848 C7JH8N 155552861 IC50 > 20000 nM T37848 C0ASJ7 155553201 IC50 = 3600 nM T37848 CUH7R2 155553391 IC50 > 10000 nM T37848 C7JCS2 155553955 IC50 < 10000 nM T37848 C0JV5A 155554027 IC50 = 2511.89 nM T37848 C7N5HA 155554052 IC50 = 16400 nM T37848 C3J2YD 155554863 IC50 = 900 nM T37848 C3Z4QS 155554969 IC50 = 17200 nM T37848 C8Q2FG 155555556 IC50 > 20000 nM T37848 C09FGY 155555863 IC50 < 10000 nM T37848 CIK75H 155556042 IC50 > 25000 nM T37848 CH0QI2 155556200 IC50 > 25000 nM T37848 C3WT2Q 155556441 IC50 > 50000 nM T37848 C9H1VK 155556442 IC50 > 50000 nM T37848 CQ3YK6 155556791 IC50 > 25000 nM T37848 CEW5U4 155556807 IC50 > 50118.72 nM T37848 CQB48L 155556931 IC50 > 50000 nM T37848 CFS63H 155557182 IC50 = 13000 nM T37848 CNH27R 155557555 IC50 = 16700 nM T37848 CPS43I 155557577 IC50 > 10000 nM T37848 C7HFI8 155558403 IC50 > 100000 nM T37848 CR70CB 155558458 IC50 < 1000 nM T37848 C4HPK2 155558743 IC50 > 25000 nM T37848 C2OJS0 155558755 IC50 = 3162.28 nM T37848 CUI6H0 155558903 IC50 > 25000 nM T37848 CKZT21 155559364 IC50 > 20000 nM T37848 C2AGR5 155559542 IC50 = 7600 nM T37848 CTI7O1 155559782 IC50 > 10000 nM T37848 CEF9N6 155560028 IC50 < 10000 nM T37848 CW2N7D 155560551 IC50 = 1100 nM T37848 C1NVA6 155560651 IC50 > 30000 nM T37848 CF4LM6 155560880 IC50 > 25000 nM T37848 C9GM1C 155561039 IC50 > 10000 nM T37848 CM7ZG9 155561160 IC50 = 10000 nM T37848 C9HIU5 155561551 IC50 < 10000 nM T37848 C1MW3L 155561646 IC50 > 40000 nM T37848 CO03PN 155561762 IC50 = 251.5 nM T37848 CALB48 155561861 IC50 > 10000 nM T37848 CL3A2S 155562076 IC50 = 100 nM T37848 CKX10W 155562129 IC50 > 50000 nM T37848 C6T2RV 155562253 IC50 < 10000 nM T37848 CCOD50 155562467 IC50 = 2230 nM T37848 CFVB79 155562854 IC50 = 40000 nM T37848 CAB5U7 155562903 IC50 > 25000 nM T37848 CWM03V 155563050 IC50 > 39810.72 nM T37848 CG95WV 155563831 IC50 > 20000 nM T37848 CXEW19 155563979 IC50 > 25000 nM T37848 CWOE21 155564042 IC50 > 30000 nM T37848 CZ6TP2 155564129 IC50 > 10000 nM T37848 CZR6W0 155564401 IC50 > 10000 nM T37848 CAZM60 155564535 IC50 = 25118.86 nM T37848 CMK03D 155564568 IC50 < 10000 nM T37848 CC5FE7 155564581 IC50 > 50000 nM T37848 CMR8A9 155565213 IC50 > 10000 nM T37848 C63GJB 155567000 IC50 > 25000 nM T37848 C37BGO 155567311 IC50 > 30000 nM T37848 C08ZCY 155567532 IC50 > 50000 nM T37848 CO58ME 155567694 IC50 = 1600 nM T37848 CK9N0Z 155567885 IC50 > 10000 nM T37848 CMC2A9 155568311 IC50 > 50000 nM T37848 C5GXM4 155569310 IC50 > 50000 nM T37848 C94IJB 10367131 IC50 = 10000 nM T37848 C0T4GZ 136166859 IC50 < 200 nM T37848 CK6VX4 136166933 IC50 < 200 nM T37848 CYIU14 16750228 IC50 = 2800 nM T37848 CI67WG 16750292 IC50 = 2500 nM T37848 C9JX2G 53363150 IC50 = 370 nM T37848 CU76JB 53363338 IC50 > 10000 nM T37848 CI8LX0 57976125 IC50 = 26000 nM T37848 CKYJ21 76283430 IC50 > 20000 nM T37848 CIJ3N0 76283682 IC50 > 30000 nM T37848 D00AEX 44341439 IC50 = 76900 nM T37848 D00AWM 9826520 IC50 = 1600 nM T37848 D00DSE 49864196 IC50 = 668 nM T37848 D00EMF 3644637 IC50 > 100000 nM T37848 D00GOQ 44575384 IC50 = 7700 nM T37848 D00PYW 44341256 IC50 = 5670 nM T37848 D00TOF 193042 Ki = 142 nM T37848 D00XDG 11708263 IC50 > 30000 nM T37848 D00YEV 5281605 IC50 = 9200 nM T37848 D00YNA 25093374 IC50 = 800 nM T37848 D01ARE 44388719 IC50 = 6300 nM T37848 D01FBL 442835 Ki = 177 nM T37848 D01JFF 44191096 IC50 > 30000 nM T37848 D01JPJ 66731056 IC50 > 10000 nM T37848 D01JXM 46222048 IC50 = 470 nM T37848 D01REI 46901610 IC50 = 7580 nM T37848 D01RZP 25192621 IC50 = 1500 nM T37848 D01UYI 5281607 IC50 > 50000 nM T37848 D01YWE 25207521 IC50 > 10000 nM T37848 D02BGR 9949648 IC50 = 22000 nM T37848 D02DEF 49765871 IC50 > 30000 nM T37848 D02DTR 44341278 IC50 = 417 nM T37848 D02EAP 11993867 Ki = 1100 nM T37848 D02GFK 25034431 IC50 = 21070 nM T37848 D02HNQ 46182736 IC50 > 25000 nM T37848 D02HSP 44575401 IC50 = 15000 nM T37848 D02KZD 71598521 IC50 = 16000 nM T37848 D02SGJ 19009 IC50 = 900 nM T37848 D02TKC 10429288 Ki = 10000 nM T37848 D02TSN 46244454 IC50 > 10000 nM T37848 D02YNH 9901086 IC50 > 50000 nM T37848 D03DMA 44429171 IC50 = 42930 nM T37848 D03EXD 49864181 IC50 = 3210 nM T37848 D03KXT 44341260 IC50 = 344 nM T37848 D03MUZ 17759555 IC50 = 9000 nM T37848 D03NMM 46843035 IC50 = 8800 nM T37848 D03YHZ 25147692 IC50 < 50000 nM T37848 D04ISG 11680597 IC50 = 3560 nM T37848 D04VPH 45376872 IC50 > 30000 nM T37848 D05KIF 13916150 IC50 = 14900 nM T37848 D05LKO 44414722 IC50 = 194000 nM T37848 D05MSG 44593666 IC50 = 26000 nM T37848 D05NWH 443390 IC50 = 9000 nM T37848 D05UZY 11539096 IC50 = 23500 nM T37848 D05VQJ 25147749 IC50 > 10000 nM T37848 D05XGR 6918647 IC50 = 6000 nM T37848 D06CWR 24754344 IC50 = 3540 nM T37848 D06DSX 12304178 IC50 = 13400 nM T37848 D06EMC 11392888 IC50 > 30000 nM T37848 D06HOI 44249821 IC50 = 18500 nM T37848 D06MBD 11176403 IC50 = 3860 nM T37848 D06MLU 332806 Ki = 54 nM T37848 D06QFO 11332763 Ki = 23600 nM T37848 D06TRS 23646069 Ki = 3000 nM T37848 D06UEP 17027464 IC50 = 20900 nM T37848 D06VDN 443391 IC50 > 100000 nM T37848 D07ADX 54764565 IC50 = 16200 nM T37848 D07ANY 1367 IC50 = 450 nM T37848 D07GCA 11514705 IC50 > 10000 nM T37848 D07VGT 46901929 IC50 = 1140 nM T37848 D07VHB 11321889 IC50 = 348 nM T37848 D07WLT 25180108 IC50 = 6210 nM T37848 D08BOH 192827 IC50 = 1100 nM T37848 D08FZC 161373 IC50 = 1000 nM T37848 D08IDC 24827305 IC50 = 1913 nM T37848 D08QPU 72737723 IC50 = 15600 nM T37848 D08TSE 44191463 Ki = 158.49 nM T37848 D08UWZ 16725047 IC50 > 40000 nM T37848 D08XVZ 24866313 IC50 = 5700000 nM T37848 D08ZYC 11595431 IC50 > 33000 nM T37848 D09ALJ 5280805 IC50 > 80000 nM T37848 D09CPC 13728862 IC50 = 127000 nM T37848 D09PTP 57325421 IC50 > 10000 nM T37848 D09REF 443672 Ki = 7600 nM T37848 D09VMS 44575398 Ki = 82 nM T37848 D09VTJ 441298 IC50 = 2300 nM T37848 D09YEQ 11158623 IC50 = 4800 nM T37848 D09ZPN 135416394 IC50 > 100000 nM T37848 D0A0GU 44247568 IC50 > 10000 nM T37848 D0A1SJ 44575400 IC50 = 440 nM T37848 D0AS0V 10141 IC50 > 10000 nM T37848 D0B0LC 44341428 IC50 = 630 nM T37848 D0B2ZB 3013841 IC50 = 7400 nM T37848 D0BD6A 10278617 IC50 = 5300 nM T37848 D0BU8W 44219611 IC50 > 100000 nM T37848 D0BV3B 16214871 IC50 > 30000 nM T37848 D0C2GE 67161540 IC50 > 50000 nM T37848 D0D5YP 5280371 IC50 = 24920 nM T37848 D0DA1E 23642319 IC50 > 10000 nM T37848 D0DY5G 443389 IC50 > 100000 nM T37848 D0E2GV 44191462 Ki = 251.19 nM T37848 D0F5EI 10017019 IC50 > 10000 nM T37848 D0G6BJ 24802842 IC50 = 10000 nM T37848 D0G9WP 18407230 IC50 < 200000 nM T37848 D0G9YL 16214849 IC50 = 4600 nM T37848 D0H1OK 11562302 IC50 = 62000 nM T37848 D0I1YH 46901446 IC50 = 538 nM T37848 D0I7GE 11790 IC50 > 10000 nM T37848 D0I9PF 60182322 IC50 = 38 nM T37848 D0IB3K 5320686 IC50 = 700 nM T37848 D0IM5E 11450263 IC50 >= 55000 nM T37848 D0IO8J 3025961 IC50 > 100000 nM T37848 D0J0TP 9917862 IC50 > 30000 nM T37848 D0J1IE 11993873 Ki = 7400 nM T37848 D0J1QT 44473100 IC50 = 39000 nM T37848 D0J4CB 24803184 IC50 = 8000 nM T37848 D0K3EW 49799108 IC50 = 3000 nM T37848 D0K4LS 10691533 IC50 = 76032627.69 nM T37848 D0L2WP 46225540 IC50 = 50 nM T37848 D0M0IQ 11210706 IC50 > 400000 nM T37848 D0M0KX 25192477 IC50 = 820 nM T37848 D0M0QJ 10452725 IC50 = 53000 nM T37848 D0M4SY 135440466 IC50 = 500 nM T37848 D0N2KU 44517677 IC50 = 12200 nM T37848 D0N4LR 53469448 IC50 = 10000 nM T37848 D0NC3P 117443 IC50 = 9100 nM T37848 D0NC8V 6918854 IC50 = 4000 nM T37848 D0NM0P 25093389 IC50 = 1900 nM T37848 D0O1HH 11263510 Ki = 15200 nM T37848 D0O8WT 10338547 IC50 > 30000 nM T37848 D0OQ1I 72376 Ki = 630 nM T37848 D0P0IE 10205 IC50 > 10000 nM T37848 D0P8PK 10192730 IC50 = 1580 nM T37848 D0PC5A 44243144 IC50 > 10000 nM T37848 D0Q0BK 46901611 IC50 = 896 nM T37848 D0Q7QU 107917 IC50 = 10000 nM T37848 D0R0IB 56587994 IC50 > 30000 nM T37848 D0R0TW 11964036 IC50 > 10000 nM T37848 D0R2TW 10238338 IC50 = 89000 nM T37848 D0S0QN 1712706 IC50 = 5105050 nM T37848 D0S6GE 5327067 IC50 = 25000 nM T37848 D0S6NP 5280862 IC50 = 36200 nM T37848 D0S9CI 11989776 IC50 > 30000 nM T37848 D0T4AC 11259008 IC50 = 830 nM T37848 D0U7BJ 44341234 IC50 = 252 nM T37848 D0U7OD 16043230 IC50 = 30000 nM T37848 D0V0NM 72323 IC50 = 2100 nM T37848 D0V0YM 24871527 IC50 = 3300 nM T37848 D0V2QH 24894072 IC50 = 2770 nM T37848 D0V3ZG 25192022 IC50 > 7500 nM T37848 D0V4EX 54760053 IC50 > 40000 nM T37848 D0VD5O 11148236 Ki = 19600 nM T37848 D0W3XD 16049828 IC50 = 12000 nM T37848 D0WN9P 46901444 IC50 = 1520 nM T37848 D0WU1S 52912189 IC50 = 9700 nM T37848 D0X3CF 442879 Ki = 373 nM T37848 D0Y1YR 442793 IC50 = 21800 nM T37848 D0Y2RL 25192475 IC50 = 500 nM T37848 D0Y4BL 11676971 IC50 = 4800 nM T37848 D0Y5KX 46901443 IC50 = 2450 nM T37848 D0YM4A 22319604 IC50 > 10000 nM T37848 D0YP4A 11993866 Ki = 3100 nM T37848 D0YQ8U 11993871 Ki = 63000 nM T37848 D0YQ8V 46236221 IC50 > 30000 nM T37848 D0YW6B 44627267 IC50 = 16700 nM T37848 D0Z7TM 22273644 IC50 = 11500 nM T37848 D0ZY7X 697226 IC50 > 5000 nM T09022 D00UVA 11556711 IC50 = 620 nM T09022 D0SH3I 387447 IC50 = 940 nM T09022 D0DP0J 92135659 IC50 > 10000 nM T09022 D0VO0T 24800541 IC50 = 10 nM T09022 CLU69K 10628969 IC50 = 8000 nM T09022 CU0FE7 24752894 IC50 = 25000 nM T09022 CEV5D1 49859748 IC50 = 34000 nM T09022 C82JTA 71305068 IC50 = 27200 nM T09022 C45HOE 71562349 IC50 = 20 nM T09022 CGY43C 78425867 IC50 > 25000 nM T09022 CC0OF1 101874274 IC50 = 410 nM T09022 CG0N1O 101874275 IC50 > 10000 nM T09022 CL50TR 101874276 IC50 > 10000 nM T09022 C0RY3V 101874277 IC50 > 10000 nM T09022 CVHC29 101874278 IC50 > 100000 nM T09022 C4VHU6 101874279 IC50 > 10000 nM T09022 C9C5OZ 117607839 IC50 > 25000 nM T09022 CLHS74 117607901 IC50 = 1437 nM T09022 CW9R0U 117607904 IC50 = 0.131 nM T09022 C7QST8 117611788 IC50 > 250000 nM T09022 CO1HJ9 117611880 IC50 > 250000 nM T09022 C9YH1X 117611941 IC50 > 250000 nM T09022 C0WZ3V 118709677 IC50 > 100000 nM T09022 C14VLB 118709678 IC50 > 30000 nM T09022 CO5CU1 118709679 IC50 > 100000 nM T09022 C1RA9C 118709680 IC50 > 100000 nM T09022 CL45BO 145960456 IC50 = 210 nM T09022 C5G6LM 145961320 IC50 = 130 nM T09022 CUIF27 145961566 IC50 = 1110 nM T09022 CI9JH6 145961877 IC50 = 400 nM T09022 C3M4OD 145961898 IC50 = 395 nM T09022 C8CSZ0 145962247 IC50 = 360 nM T09022 C97URS 145962850 IC50 = 200 nM T09022 COA19G 145963426 IC50 = 300 nM T09022 CM3D8G 145979576 IC50 = 79000 nM T09022 CEI3U1 145979850 IC50 = 16000 nM T09022 C5AYC4 145980811 IC50 = 106000 nM T09022 C41IRV 145981707 IC50 = 14300 nM T09022 C5X3GQ 145986425 IC50 = 8900 nM T09022 CM3H4F 145987197 IC50 = 820 nM T09022 CNZ7R6 145987536 IC50 = 21400 nM T09022 CV1D7O 145987617 IC50 = 22000 nM T09022 C1EF3B 145988020 IC50 = 6600 nM T09022 CE16JH 145989568 IC50 = 28300 nM T09022 CXG30R 145990249 IC50 = 30000 nM T09022 CBY18W 145992498 IC50 = 2700 nM T09022 CJO08K 145993925 IC50 = 5800 nM T09022 C5AUF0 155510519 IC50 = 22 nM T09022 C2O9TA 155511183 IC50 = 200 nM T09022 C2NW8K 155511747 IC50 = 6400 nM T09022 CBHD46 155513331 IC50 = 850 nM T09022 C8E6ZX 155514792 IC50 = 230 nM T09022 CH0BW8 155514969 IC50 = 2300 nM T09022 CIS75B 155515280 IC50 = 915 nM T09022 C53ZEN 155516179 IC50 = 3100 nM T09022 CM3BV8 155516620 IC50 = 34000 nM T09022 CHR3P8 155517182 IC50 = 48040 nM T09022 C6OM9X 155517411 IC50 = 170 nM T09022 CEW35H 155518001 IC50 > 10000 nM T09022 CE95IQ 155518158 IC50 = 180 nM T09022 CU6N7M 155518236 IC50 = 420 nM T09022 CJLN49 155519553 IC50 = 230 nM T09022 CM74XQ 155520942 IC50 = 204 nM T09022 CNM0Q9 155521286 IC50 = 420 nM T09022 CZKF54 155521690 IC50 = 140 nM T09022 C8GNQ9 155522828 IC50 = 71 nM T09022 CW75YK 155523151 IC50 > 100000 nM T09022 CWU6I8 155524626 IC50 = 350 nM T09022 CK8P7I 155524958 IC50 = 61 nM T09022 CNVG12 155526191 IC50 = 47 nM T09022 CW8K6C 155527076 IC50 = 200 nM T09022 C3VF1Y 155528807 IC50 = 4250 nM T09022 C6C5BW 155529708 IC50 = 280 nM T09022 C8LK5P 155529890 IC50 > 10000 nM T09022 C65BEV 155530124 IC50 = 350 nM T09022 C3BK1V 155530730 IC50 = 175 nM T09022 CUP2B4 155531358 IC50 = 97 nM T09022 CGX87Q 155531944 IC50 = 260 nM T09022 C9JCR8 155533457 IC50 > 10000 nM T09022 C2MTK4 155534927 IC50 = 39 nM T09022 CZ7FR4 155534939 IC50 = 106 nM T09022 C2NTI6 155538936 IC50 = 159 nM T09022 CO70SA 155539427 IC50 = 45 nM T09022 C6OIY3 155541618 IC50 = 2500 nM T09022 CY2TS3 155546980 IC50 = 1350 nM T09022 C8ELR3 155547121 IC50 > 10000 nM T09022 CL6MV8 155549641 IC50 = 97 nM T09022 CID4F3 155550143 IC50 > 10000 nM T09022 CS0FV9 155550266 IC50 = 4100 nM T09022 C61HCU 155550509 IC50 = 23 nM T09022 CKON12 155551453 IC50 = 325 nM T09022 CSD63L 155551642 IC50 = 130 nM T09022 CBHM14 155553205 IC50 = 380 nM T09022 C35NJC 155553210 IC50 > 1000 nM T09022 CI15FC 155553565 IC50 = 2500 nM T09022 CVJ3E7 155553910 IC50 = 57 nM T09022 C6YP0L 155554916 IC50 = 12000 nM T09022 CJX84Z 155555024 IC50 = 47 nM T09022 CA1GX2 155560146 IC50 = 700 nM T09022 COV3C6 155560154 IC50 = 1150 nM T09022 C0DYR3 155561372 IC50 > 10000 nM T09022 CB17JR 155561390 IC50 > 10000 nM T09022 C5Z7YC 155567712 IC50 = 110 nM T09022 C84ZYD 155568489 IC50 = 360 nM T09022 C4ZV3Q 155568941 IC50 = 2900 nM T09022 D0Q4MO 23642227 IC50 = 590 nM T78915 CX04HL 736190 IC50 > 100000 nM T78915 CXC69A 16678113 IC50 = 26 nM T78915 CPO5K4 23633257 IC50 = 70 nM T78915 C7BPJ5 23633323 IC50 > 11000 nM T78915 C7SK4I 23633324 IC50 = 200 nM T78915 CY4E2S 23633464 IC50 = 380 nM T78915 CKN64Y 23634107 IC50 = 890 nM T78915 CHSE14 23634109 IC50 > 10000 nM T78915 CEG51A 23634331 IC50 = 32 nM T78915 CJ8SK0 24894403 IC50 = 240 nM T78915 C9FBJ0 24894404 IC50 = 960 nM T78915 CLPM54 24894405 IC50 = 110 nM T78915 CN14DF 24894499 IC50 = 6150 nM T78915 CF45MO 24894500 IC50 = 190 nM T78915 CKVI72 24894501 IC50 = 46 nM T78915 CE4G8Y 24894502 IC50 = 13 nM T78915 CU01MS 24894503 IC50 = 31 nM T78915 CI7JL3 24894504 IC50 = 69 nM T78915 CCIK07 24894612 IC50 = 44 nM T78915 CLE08X 24894613 IC50 = 40 nM T78915 CB0D5A 24894617 IC50 = 770 nM T78915 C8SUE3 24894758 IC50 = 12600 nM T78915 CH9K4C 24894759 IC50 = 24 nM T78915 CK6N2D 24894761 IC50 = 29 nM T78915 C46PBE 24894881 IC50 = 11100 nM T78915 CN94LG 24894987 IC50 = 970 nM T78915 CN38OI 24894988 IC50 > 10000 nM T78915 CJ9YM8 24894989 IC50 = 180 nM T78915 CZBX15 24894990 IC50 = 24 nM T78915 CHS29V 25025298 IC50 = 16 nM T78915 CDKB49 25144187 IC50 = 19 nM T78915 C40LZS 25153819 IC50 = 14 nM T78915 CV83LS 25153820 IC50 = 15600 nM T78915 COT12L 44560453 IC50 = 45 nM T78915 C7E0NA 44560934 IC50 = 3770 nM T78915 C5CMV4 44560969 IC50 = 54 nM T78915 CF40HI 45486488 IC50 = 7 nM T78915 CV70IP 45486489 IC50 = 44 nM T78915 CHVB76 45486494 IC50 = 38 nM T78915 C7T8DR 45486495 IC50 = 150 nM T78915 CG4OB9 45486500 IC50 = 250 nM T78915 CD8M3P 45486509 IC50 = 55 nM T78915 C9DOM3 45486510 IC50 = 610 nM T78915 C01WNH 45486518 IC50 = 190 nM T78915 C15XUM 45486538 IC50 = 160 nM T78915 CQ4IY7 45486543 IC50 = 24 nM T78915 CNY0B6 45486544 IC50 = 320 nM T78915 C1LDS0 45486548 IC50 = 500 nM T78915 CTW1V7 45486562 IC50 = 120 nM T78915 CMS5A1 45486563 IC50 = 100 nM T78915 CNO42T 45486568 IC50 = 120 nM T78915 CJH81F 45486569 IC50 = 330 nM T78915 C10LZN 45486570 IC50 = 50 nM T78915 C7T2SU 45486578 IC50 = 60 nM T78915 CQMV97 45486579 IC50 = 150 nM T78915 CV4O9M 45486580 IC50 = 120 nM T78915 C6X9RN 117942064 IC50 = 55 nM T78915 CHJ2V9 117942361 IC50 = 26 nM T78915 C90HKB 117942565 IC50 = 30 nM T78915 CY7MN5 117943003 IC50 = 77 nM T78915 C4Y6HN 117947646 IC50 = 20 nM T78915 CL2BP0 117947705 IC50 = 33 nM T78915 CY03DN 117947820 IC50 = 2266 nM T78915 C89ZQD 117951704 IC50 = 32 nM T78915 C1YK4U 117951765 IC50 = 35 nM T78915 CO4Q3E 117951768 IC50 = 79 nM T78915 CY3PK8 117951788 IC50 = 1125 nM T78915 C6ZO2V 117951880 IC50 = 14 nM T78915 CTC65B 117951917 IC50 = 949 nM T78915 CDC4O1 117951922 IC50 = 30 nM T78915 C6F4NE 117951942 IC50 = 25 nM T78915 CZH7Q1 117952010 IC50 = 39 nM T78915 C0YL5C 117952014 IC50 = 28 nM T78915 C15MHC 117952015 IC50 = 40 nM T78915 C1BY5Q 117952041 IC50 = 26 nM T78915 C0A4OP 117952075 IC50 = 51 nM T78915 C3PYL2 117952130 IC50 = 23 nM T78915 CC3AH2 117952139 IC50 = 128 nM T78915 C31UCV 117952142 IC50 = 1787 nM T78915 CW9VO3 117952156 IC50 = 62 nM T78915 C0C3FQ 117952261 IC50 = 32 nM T78915 CM3TX5 117952268 IC50 = 11 nM T78915 CM21FS 117952298 IC50 = 211 nM T78915 CPD8Z1 117952310 IC50 = 21 nM T78915 C1LE6D 117952313 IC50 = 53 nM T78915 C0E4BH 117952436 IC50 = 207 nM T78915 CI3Z7K 117952506 IC50 = 65 nM T78915 CIM5F2 117952561 IC50 = 26 nM T78915 C25LPC 117952603 IC50 = 73 nM T78915 CQ14LK 117952608 IC50 = 37 nM T78915 C6EZ4I 117952632 IC50 = 65 nM T78915 CA2VT9 117952644 IC50 = 23 nM T78915 C9ROG8 117952675 IC50 = 40 nM T78915 CZW6E9 117952688 IC50 = 5930 nM T78915 C3O2RZ 117952705 IC50 = 885 nM T78915 C6XEA1 117952772 IC50 = 35 nM T78915 C4CTY1 117952796 IC50 = 53 nM T78915 C2YMC1 117952807 IC50 = 32 nM T78915 C65ZUJ 117952825 IC50 = 19 nM T78915 C5PSG1 117952837 IC50 = 30 nM T78915 CH8KW6 117952867 IC50 = 22 nM T78915 CZF78T 117952886 IC50 = 22 nM T78915 CVT1G8 118138444 IC50 = 22 nM T78915 C92EFA 118138451 IC50 = 15 nM T78915 C2UHI8 118138452 IC50 = 18 nM T78915 C71GFP 118138453 IC50 = 32 nM T78915 CM8K1C 118138476 IC50 = 30 nM T78915 C8AER7 118138477 IC50 = 61 nM T78915 CPK74Z 118138494 IC50 = 35 nM T78915 CV3H5W 118138498 IC50 = 7 nM T78915 CG2HL8 118138501 IC50 = 2200 nM T78915 CYU9J2 118138508 IC50 = 16 nM T78915 CD7YT3 118138513 IC50 = 599 nM T78915 C70SZE 118138529 IC50 = 38 nM T78915 C9K7IO 118138537 IC50 = 14 nM T78915 C7R0IK 118138541 IC50 = 74 nM T78915 CPZM24 118138545 IC50 = 66 nM T78915 CC0Z6Y 118138548 IC50 = 11 nM T78915 CB70CG 118138559 IC50 = 20 nM T78915 CSGT89 118138585 IC50 = 99 nM T78915 C6L8BP 118138593 IC50 = 11036 nM T78915 CEL32W 118138597 IC50 = 15 nM T78915 C8YH4U 118138600 IC50 = 26 nM T78915 CRQF14 118138608 IC50 = 22 nM T78915 C72RFA 118138612 IC50 = 10 nM T78915 C53LFO 118138613 IC50 = 8 nM T78915 CL0OS8 118138618 IC50 = 58 nM T78915 C60SCL 118138641 IC50 = 106 nM T78915 C3SD8Q 118138643 IC50 = 25 nM T78915 CBIQ04 118138650 IC50 = 405 nM T78915 CO9GT1 118138652 IC50 = 61 nM T78915 C84KAH 118138653 IC50 = 6 nM T78915 C3GSU1 118138655 IC50 = 46 nM T78915 CP7Y2O 118138658 IC50 = 25 nM T78915 CA0JM3 118138659 IC50 = 6 nM T78915 CM02PW 118138660 IC50 = 165 nM T78915 C7QIC4 118138662 IC50 = 11 nM T78915 C50SVU 118138667 IC50 = 43 nM T78915 CV71QZ 118138668 IC50 = 129 nM T78915 C17PXI 118138675 IC50 = 28 nM T78915 C6JA0I 118138679 IC50 = 11 nM T78915 CTL23M 118138682 IC50 = 11 nM T78915 CC9KJ4 118138687 IC50 = 16 nM T78915 C7QRI0 118138690 IC50 = 106 nM T78915 C1GDL3 118138692 IC50 = 33 nM T78915 C8IE2K 118138697 IC50 = 1844 nM T78915 CG5Y7M 118138698 IC50 = 6 nM T78915 COE9A4 118138701 IC50 = 16 nM T78915 CL6G5A 118138702 IC50 = 13 nM T78915 C4Z7OX 118138709 IC50 = 15 nM T78915 C7EO1T 118138727 IC50 = 666 nM T78915 CN24DU 118138728 IC50 = 33 nM T78915 CI1M9K 118138734 IC50 = 5107 nM T78915 C2W3MV 118138743 IC50 = 53 nM T78915 CJ74ZI 118138748 IC50 = 14 nM T78915 CI7L2R 118138786 IC50 = 10 nM T78915 CB7WY5 118138788 IC50 = 12 nM T78915 CN52GV 118138797 IC50 = 54 nM T78915 CES12W 118138805 IC50 = 45 nM T78915 CNC07L 118138814 IC50 = 69 nM T78915 CNG53H 118138822 IC50 = 335 nM T78915 C57HKU 127027748 IC50 = 50 nM T78915 CYG0L2 127027749 IC50 = 96 nM T78915 CL39CP 127027750 IC50 = 211 nM T78915 C6IFG3 127039050 IC50 = 361 nM T78915 CYX75V 127039051 IC50 = 449 nM T78915 C8IBL6 127039363 IC50 = 583 nM T78915 CZA72X 127040033 IC50 = 519 nM T78915 C3QFO0 127040034 IC50 = 1019 nM T78915 COZ38I 127040365 IC50 = 1050 nM T78915 C2LW9R 127040366 IC50 = 1355 nM T78915 C38XSZ 127040686 IC50 = 2961 nM T78915 CDJL87 127040687 IC50 = 3422 nM T78915 C83KIB 127040688 IC50 = 20000 nM T78915 C02GNB 127041032 IC50 = 1407 nM T78915 CM17CP 127041039 IC50 = 2714 nM T78915 C7E4YD 127041040 IC50 = 4039 nM T78915 CO0YL1 127041041 IC50 = 5126 nM T78915 C0WJT2 127041042 IC50 = 5257 nM T78915 C72MRB 127041043 IC50 = 6220 nM T78915 C43KME 127041339 IC50 = 871 nM T78915 CYX82H 127041340 IC50 = 1511 nM T78915 CL7W0Q 127041341 IC50 = 2149 nM T78915 CERF20 127041364 IC50 = 7552 nM T78915 CC0UP9 127041658 IC50 = 8536 nM T78915 CAQ85X 127041659 IC50 = 20000 nM T78915 C3SQ5O 127041660 IC50 = 20000 nM T78915 C53FNL 127045723 IC50 = 2014 nM T78915 CBQ38U 127046894 IC50 = 34 nM T78915 CM5U0Y 127047021 IC50 = 501 nM T78915 CS3E1B 127047046 IC50 = 19 nM T78915 CVU69N 127047215 IC50 = 20000 nM T78915 CD7Y4E 136927832 IC50 = 974 nM T78915 CR03WS 137635628 IC50 = 460 nM T62193 C2NP1D 4501 IC50 = 1340000 nM T62193 C43DAY 68635 IC50 = 200000 nM T62193 CY94ZF 149257 IC50 = 400000 nM T62193 CRBX80 21144709 IC50 = 3500000 nM T62193 CN7A9I 71524055 IC50 = 190000 nM T62193 CFH43U 71524058 IC50 = 1170000 nM T62193 C8MZ4F 71524092 IC50 = 120000 nM T62193 C2PD3T 90643936 IC50 = 2690000 nM T62193 C1AUE2 90643938 IC50 = 1390000 nM T62193 C7DJ6E 90643940 IC50 = 1490000 nM T62193 CD4Q1B 90643942 IC50 = 950000 nM T62193 CZ09BP 90643944 IC50 = 570000 nM T62193 CL9W0B 90643946 IC50 = 930000 nM T62193 C7I8JE 90643948 IC50 = 600000 nM T62193 D0T9ZL 2703 IC50 = 1280000 nM T06093 D04LVK 57379345 IC50 = 1270 nM T06093 D0B5LF 448042 Ki = 300 nM T06093 D0EG1I 9926791 IC50 = 3400 nM T06093 D01ZAQ 25227436 IC50 = 56 nM T06093 D02ZQS 16095342 IC50 = 4 nM T06093 D03KKR 3547 IC50 = 158 nM T06093 D03LWG 53235510 IC50 > 10000 nM T06093 D07EHV 44814409 IC50 > 10000 nM T06093 D08ZPO 448043 IC50 = 5 nM T06093 D09XZL 56962369 IC50 = 10 nM T06093 D0E3TC 44259 IC50 = 0.933 nM T06093 D0U5UC 11950170 IC50 = 100 nM T06093 D0U9LT 9810884 IC50 = 58 nM T06093 D03BNU 59604787 IC50 > 10000 nM T06093 D0CW9Q 56596554 IC50 = 670 nM T06093 D0T3ME 156422 IC50 > 30000 nM T06093 C8BZK3 5711 IC50 = 140 nM T06093 CWI59L 88012 IC50 = 119700 nM T06093 CF7VJ0 883549 IC50 > 10000 nM T06093 CLJ97Z 963518 IC50 = 1900 nM T06093 C86HDP 1959269 IC50 > 10000 nM T06093 C49YTC 2227730 IC50 = 357200 nM T06093 CT7L1J 2766553 IC50 = 1700 nM T06093 CIU9K1 3049109 IC50 = 55900 nM T06093 CHF4O5 4356253 IC50 = 590 nM T06093 CZX36A 4421488 IC50 = 61800 nM T06093 CEU1N6 5056270 IC50 = 0.56 nM T06093 CI26XO 6910830 IC50 = 7400 nM T06093 C4TJ9V 9579814 IC50 = 640 nM T06093 CA80PO 9661728 IC50 = 300 nM T06093 CO08EA 9714186 IC50 = 3700 nM T06093 CEB53H 9724880 IC50 = 62 nM T06093 C4KEJ2 9860439 IC50 = 390 nM T06093 CV50OB 9863672 IC50 = 3.8 nM T06093 CM5Z8X 9869943 IC50 > 1000 nM T06093 C9O3XQ 9901617 IC50 = 61 nM T06093 C2Y3WG 9907612 IC50 = 14000 nM T06093 CJO47T 9948405 IC50 > 10000 nM T06093 CB76YH 9994431 IC50 > 100000 nM T06093 CV8I5X 9999342 IC50 > 10000 nM T06093 C1B0RN 10014369 IC50 = 1300 nM T06093 C5TQ7X 10247543 IC50 > 10000 nM T06093 C7SFI1 10296883 IC50 > 10000 nM T06093 C2WQ8M 10473563 IC50 > 10000 nM T06093 C48HIZ 11155477 IC50 = 190 nM T06093 CR6U2M 11196984 IC50 = 120 nM T06093 CBOP58 11293798 Ki > 10000 nM T06093 C26BZX 11362471 Ki > 10000 nM T06093 C43NPS 11373886 IC50 > 10000 nM T06093 CWXB93 11397177 Ki > 10000 nM T06093 C0APW4 11422034 IC50 = 10000 nM T06093 CQR05P 11494718 IC50 = 24 nM T06093 C0H6QS 11495680 IC50 > 10000 nM T06093 CHT93E 11502159 IC50 = 23 nM T06093 CIW9L5 11502867 IC50 > 10000 nM T06093 CEK1G9 11503627 IC50 = 6300 nM T06093 C5FMJ4 11507964 Ki = 2.3 nM T06093 CK2Q0X 11516978 IC50 > 10000 nM T06093 CNQ61U 11524891 IC50 = 1900 nM T06093 CPE53F 11526238 IC50 > 10000 nM T06093 CE9R7D 11530100 IC50 = 58000 nM T06093 C5BM4T 11531799 IC50 > 10000 nM T06093 C53OSD 11532048 IC50 > 10000 nM T06093 CC4QM5 11532676 IC50 > 10000 nM T06093 CXL01N 11536733 IC50 = 53000 nM T06093 CR92GA 11537005 IC50 = 21 nM T06093 CTG83F 11539329 Ki > 7500 nM T06093 C01FVM 11546457 IC50 > 10000 nM T06093 CME81U 11560302 IC50 = 950 nM T06093 CN08CJ 11561907 IC50 = 220 nM T06093 CNBM81 11562171 IC50 > 10000 nM T06093 CUW0C5 11567501 IC50 = 30 nM T06093 CWRY72 11567821 IC50 = 20 nM T06093 CO9KP5 11583459 IC50 > 5000 nM T06093 CMIL86 11590363 Ki > 7500 nM T06093 C0NV9Y 11596881 IC50 > 10000 nM T06093 C4WCL9 11603404 IC50 = 18 nM T06093 CJ5K9X 11609495 IC50 = 530 nM T06093 C6LDN4 11617898 IC50 = 60 nM T06093 C1BLZ5 11620055 IC50 > 10000 nM T06093 C9T6SC 11640926 Ki > 7500 nM T06093 C24GRQ 11661959 IC50 > 10000 nM T06093 CQGI52 11667631 IC50 = 2500 nM T06093 C0V7SU 11675388 IC50 = 66 nM T06093 CS72ED 11682843 IC50 > 10000 nM T06093 CJ9KN7 11683817 IC50 > 10000 nM T06093 CU0E8O 11690457 Ki < 4 nM T06093 CLC53E 11691173 IC50 > 10000 nM T06093 CXS4V3 11694866 IC50 = 2500 nM T06093 C43TXY 11703935 IC50 > 10000 nM T06093 C6AH2S 11716019 IC50 = 2900 nM T06093 C1FTX3 11719305 IC50 > 10000 nM T06093 CFPW41 16007116 Ki > 7500 nM T06093 C9TU1O 16046126 IC50 > 1000 nM T06093 C7WZY3 16066456 IC50 = 94 nM T06093 C7Z4LV 16095343 IC50 = 7 nM T06093 C54YXC 16121514 IC50 = 2.455 nM T06093 CZF23I 16124479 IC50 = 38.9 nM T06093 C5VPH9 16129448 IC50 = 248 nM T06093 CY09ZD 16219471 IC50 = 508.8 nM T06093 CS8W9L 16222361 IC50 = 91.2 nM T06093 CA20NM 16222570 IC50 = 1122.02 nM T06093 C9M0IS 16662085 IC50 = 10000 nM T06093 C5AB3F 16662086 IC50 = 770 nM T06093 CRL96A 16662087 IC50 = 1700 nM T06093 C4L1FE 16662089 IC50 = 1200 nM T06093 CG9VH4 16662090 IC50 = 1000 nM T06093 CYJS23 16662091 IC50 = 190 nM T06093 CU0V6D 16662092 IC50 = 3900 nM T06093 C2AL3D 16662093 IC50 = 800 nM T06093 CSW16Z 16662094 IC50 = 5300 nM T06093 CR8I4H 16662096 IC50 = 100 nM T06093 C5FH6G 16662098 IC50 = 1300 nM T06093 CA2OZ7 16662100 IC50 = 190 nM T06093 C2UTD6 16662102 IC50 = 760 nM T06093 CZ9I1L 16662104 IC50 = 380 nM T06093 CUI6P9 16662106 IC50 > 10000 nM T06093 C8CIQ4 16662108 IC50 = 90 nM T06093 CS08VM 16662110 IC50 = 6000 nM T06093 C6Y1GR 16662112 IC50 = 830 nM T06093 C5O6UF 16662114 IC50 = 470 nM T06093 C9D6UT 16662116 IC50 = 150 nM T06093 CQ8U7P 16662118 IC50 = 13 nM T06093 CB21ZR 16666062 IC50 = 1.2 nM T06093 CI1J6W 16681732 IC50 = 80 nM T06093 CZT35Q 17838190 IC50 = 5500 nM T06093 CG3VB6 23646578 IC50 < 10 nM T06093 CG6D4M 23647319 IC50 > 10000 nM T06093 CY8Z7X 23647330 IC50 > 10000 nM T06093 C4XD8H 23647348 IC50 > 10000 nM T06093 CK60ZM 24758992 IC50 = 19 nM T06093 C7YG1N 24759534 IC50 = 430 nM T06093 CL59IO 24862717 IC50 = 110 nM T06093 CB4ZC7 24862718 IC50 = 845 nM T06093 C2DFH5 24863109 IC50 = 5100 nM T06093 CZ2PQ6 24863113 IC50 = 12 nM T06093 CP2I7Y 24863195 IC50 = 48 nM T06093 CZ2NR4 24863196 IC50 = 160 nM T06093 C4L1BH 24863360 IC50 = 520 nM T06093 CBYM61 24863535 IC50 = 320 nM T06093 CAJE47 24863885 IC50 = 15 nM T06093 C3KY5N 24863971 IC50 = 130 nM T06093 CR9H5B 24863972 IC50 = 35 nM T06093 CCX64S 24863973 IC50 = 120 nM T06093 C2HU6Y 24863974 IC50 = 28 nM T06093 CY8L7E 24896769 IC50 > 10000 nM T06093 CLZ23U 24951610 IC50 = 6800 nM T06093 C1ONA4 24996161 IC50 = 13 nM T06093 CX1HL8 25032704 Ki > 7500 nM T06093 CZO27W 25054032 IC50 = 69 nM T06093 CN2G3K 25054307 IC50 = 92 nM T06093 C6X5PL 25054309 IC50 = 350 nM T06093 C7EXD5 25054568 IC50 = 92 nM T06093 CNP8Q5 25054569 IC50 = 1300000 nM T06093 CRL9F4 25054571 IC50 > 6500 nM T06093 C17MSC 25054828 IC50 > 7000 nM T06093 CG82CP 25055076 IC50 = 1300 nM T06093 C7IZ6K 25055317 IC50 = 73 nM T06093 C1DNF9 25055320 IC50 = 37000 nM T06093 CFHO90 25056112 IC50 = 48 nM T06093 CV96DM 25056366 IC50 = 65000 nM T06093 CZ1KO2 25056367 IC50 = 210 nM T06093 CU8X0H 25056370 IC50 = 18 nM T06093 CV15HY 25056371 IC50 = 89 nM T06093 C0TQ1L 25056630 IC50 = 1600000 nM T06093 C76LFY 25056889 IC50 = 65 nM T06093 CS89MO 25057407 IC50 = 110000 nM T06093 CH6AU8 25057408 IC50 = 53 nM T06093 C0B7RT 25057409 IC50 = 33 nM T06093 C3AT0H 25057667 IC50 = 176 nM T06093 CJ2VI4 25057668 IC50 = 100000 nM T06093 CPST73 25057932 IC50 = 102000 nM T06093 CH7YC4 25057933 IC50 = 46 nM T06093 CM07IN 25093232 IC50 = 46 nM T06093 CZWI08 25093233 IC50 = 2 nM T06093 CV42JO 25093234 IC50 = 3.3 nM T06093 CIH3E5 25093235 IC50 = 3 nM T06093 C1S9ZE 25093236 IC50 = 920 nM T06093 CTWU37 25093237 IC50 = 760 nM T06093 C2KY1G 25094210 IC50 > 10000 nM T06093 C6BWZ8 25145145 IC50 > 100 nM T06093 C78YWA 25145716 IC50 > 500 nM T06093 CCK8D2 25154767 IC50 = 3 nM T06093 CBJ16K 25154768 IC50 < 2 nM T06093 CF0IH6 25154892 IC50 = 2 nM T06093 CB21XV 25164469 Ki = 64 nM T06093 CNF0A8 25164674 Ki = 402 nM T06093 CUX83H 25164675 Ki = 28 nM T06093 C1H7BF 25164677 Ki = 113 nM T06093 CN50EI 25164678 Ki = 822 nM T06093 C3XI7P 25164880 Ki = 1413 nM T06093 CX80QK 25164883 Ki = 6 nM T06093 C6SD2A 25165081 Ki = 315 nM T06093 C67TVH 25165085 Ki = 18 nM T06093 C8J4KL 25165278 Ki = 16 nM T06093 CRJ6M7 25165279 Ki > 6000 nM T06093 C7RBX0 25165280 Ki > 6000 nM T06093 CPEY29 25165481 Ki > 6000 nM T06093 C70DRX 25165482 Ki > 6000 nM T06093 CE8D1W 25165860 Ki = 209 nM T06093 C6VZU2 25165861 Ki = 97 nM T06093 CVI70X 25166053 Ki = 375 nM T06093 C9VA1N 25166056 Ki = 285 nM T06093 C1JS9O 25166057 Ki = 180 nM T06093 CM41PX 25166058 Ki = 285 nM T06093 CT94MS 25166059 Ki = 97 nM T06093 C5BM7F 25166250 Ki = 39 nM T06093 CCN25J 25166251 Ki = 68 nM T06093 CX8HY9 25166657 Ki = 15 nM T06093 C1CNX7 25166659 Ki = 18 nM T06093 C81WIV 25166867 Ki = 41 nM T06093 C9MR2O 25166869 Ki = 622 nM T06093 CAG1H6 25166870 Ki = 2475 nM T06093 CGUC69 25167072 Ki = 245 nM T06093 CF4G1L 25167074 Ki = 65 nM T06093 C35ZXL 25167075 Ki = 864 nM T06093 C1CRJ7 25167076 Ki = 513 nM T06093 C1IFX5 25167077 Ki = 888 nM T06093 C2D3FP 25167078 Ki = 136 nM T06093 CP2W8I 25167079 Ki = 909 nM T06093 CJO5A4 25167275 Ki = 364 nM T06093 C5KX0G 25167277 Ki = 116 nM T06093 CQ5FJ8 25167278 Ki = 1565 nM T06093 C37YSX 25167280 Ki = 226 nM T06093 C19TVC 25190767 IC50 = 977.24 nM T06093 C0CXM8 25190790 IC50 = 251.19 nM T06093 C7BAN0 25262260 IC50 = 0.7 nM T06093 CC71QJ 27666048 IC50 > 100000 nM T06093 CBQO98 42602095 IC50 = 101 nM T06093 CJ61SE 42602096 IC50 = 126 nM T06093 CI42XG 42602097 IC50 = 261 nM T06093 CD2AH4 42602175 IC50 = 76 nM T06093 CSWA85 42602176 IC50 = 89 nM T06093 C1LUN4 42602178 IC50 = 31 nM T06093 C8O3EA 42602260 IC50 = 112 nM T06093 C93NKL 42602264 IC50 = 71 nM T06093 C7WPJ5 42602351 IC50 = 37 nM T06093 C6VWM1 42629959 IC50 = 38 nM T06093 C6ND4K 43839983 IC50 = 630 nM T06093 CG4DJ2 43839997 IC50 = 280 nM T06093 CP9MW4 44124430 IC50 = 3 nM T06093 C0YHB6 44124543 IC50 = 80 nM T06093 CMAC57 44124544 IC50 = 640 nM T06093 CQ7MO2 44124778 IC50 = 78 nM T06093 C3F9EK 44124779 IC50 = 285 nM T06093 C0HB4C 44129168 IC50 < 1 nM T06093 CE7ZY8 44129169 IC50 = 6 nM T06093 CB0O2A 44186880 Ki = 230 nM T06093 C9K7OP 44186882 Ki = 108 nM T06093 CX0ZU8 44186885 Ki = 356 nM T06093 CNGV37 44189584 Ki = 635 nM T06093 CSEH15 44197303 IC50 = 7 nM T06093 C1MZF0 44197434 IC50 = 7 nM T06093 C31HWY 44197437 IC50 = 1786 nM T06093 CM8A4S 44197570 IC50 = 59 nM T06093 CA04RP 44197571 IC50 = 290 nM T06093 CR7TY6 44197572 IC50 = 51 nM T06093 CXU07O 44197573 IC50 = 10 nM T06093 CAE45R 44197710 IC50 = 15 nM T06093 CF93SL 44197978 IC50 = 17 nM T06093 CNV4P8 44198117 IC50 = 42 nM T06093 C81CXZ 44198251 IC50 = 3 nM T06093 C6WYM8 44198749 IC50 = 9 nM T06093 C1G2ZQ 44198874 IC50 = 15 nM T06093 CV09DY 44410717 IC50 > 10000 nM T06093 CP3CI1 44410720 IC50 > 10000 nM T06093 C8W7AD 44410723 IC50 > 10000 nM T06093 CAT5X4 44410829 IC50 > 10000 nM T06093 CC6Y5P 44410844 IC50 > 10000 nM T06093 CG34TY 44410851 IC50 > 10000 nM T06093 C41EIA 44410869 IC50 > 10000 nM T06093 CB6AE8 44410948 IC50 > 10000 nM T06093 CXZG12 44410949 IC50 > 10000 nM T06093 CS7IE9 44410953 IC50 > 10000 nM T06093 CA9M4X 44410954 IC50 > 10000 nM T06093 C3SP5H 44410955 IC50 > 10000 nM T06093 C5D6YP 44410956 IC50 > 10000 nM T06093 C5W1VC 44410959 IC50 > 10000 nM T06093 CM1C2G 44410960 IC50 > 10000 nM T06093 CVSI80 44411048 IC50 > 10000 nM T06093 CN72BR 44411161 IC50 > 10000 nM T06093 C4AW0O 44411183 IC50 > 10000 nM T06093 C8BAW3 44439731 IC50 = 350 nM T06093 CYH6P3 44520205 IC50 > 10000 nM T06093 CRZ79W 44542926 IC50 = 2200 nM T06093 CE0O4B 44543079 IC50 = 280 nM T06093 CQT48I 44543080 IC50 = 1100 nM T06093 C0J3GD 44562684 IC50 = 296 nM T06093 CTSU36 44562685 IC50 = 294 nM T06093 CS5WR2 44562686 IC50 = 6 nM T06093 C5DEA9 44562739 IC50 = 15 nM T06093 C2F9CI 44562740 IC50 = 78 nM T06093 CNR0X4 44562741 IC50 = 24 nM T06093 C5LJ4M 44563152 IC50 = 21 nM T06093 C5NQ8L 44563153 IC50 = 27 nM T06093 CPJ62G 44563154 IC50 = 9 nM T06093 CTN8S4 44563185 IC50 = 533 nM T06093 CQ0HI7 44563186 IC50 = 2 nM T06093 C9BWM1 44563187 IC50 = 8 nM T06093 C4RS0A 44563188 IC50 = 27 nM T06093 CE56PM 44563189 IC50 = 2 nM T06093 CH32TR 44563190 IC50 < 1 nM T06093 C05UZK 44563191 IC50 < 1 nM T06093 C6AJ5M 44571469 IC50 = 10 nM T06093 CH9Y5W 44571470 IC50 < 2 nM T06093 CQ0LO8 44571471 IC50 < 6 nM T06093 CDSA20 44571472 IC50 = 3 nM T06093 C3HUM7 44571520 IC50 = 4 nM T06093 C0XW9Q 44571521 IC50 = 4 nM T06093 C7UT4K 44571522 IC50 = 5 nM T06093 CZL8B1 44571557 IC50 = 8 nM T06093 CRSY68 44571597 IC50 = 71 nM T06093 CX1R7D 44571598 IC50 = 5 nM T06093 C1TXA9 44571599 IC50 = 4000 nM T06093 C4AF3M 44571600 IC50 = 30 nM T06093 CDCP82 44571601 IC50 = 86 nM T06093 C1KW8B 44571681 IC50 = 93 nM T06093 CR2UL3 44571682 IC50 < 6 nM T06093 CU2W7L 44571729 IC50 < 6 nM T06093 CKV96M 44571730 IC50 < 2 nM T06093 CG6P1X 44571731 IC50 = 2 nM T06093 C1WQC0 44571732 IC50 = 66 nM T06093 CCH98B 44571733 IC50 < 6 nM T06093 CI2R4A 44571777 IC50 = 12 nM T06093 CNA20Q 44571778 IC50 = 4 nM T06093 CS6C5V 44571779 IC50 < 2 nM T06093 C89HYP 44588980 IC50 = 1.5 nM T06093 CG6UW5 44634494 IC50 < 6 nM T06093 CJ0F5Q 44819015 IC50 = 2300 nM T06093 C8XH3M 44819016 IC50 > 7000000 nM T06093 CP0SB7 44819017 IC50 > 7000000 nM T06093 CLI5X3 44819018 IC50 > 7000000 nM T06093 CK5QB0 44819019 IC50 > 7000000 nM T06093 C3RNT8 44819192 IC50 = 685000 nM T06093 CN21OS 44819193 IC50 = 870 nM T06093 C7R4GT 44819194 IC50 > 7000000 nM T06093 CE7LA1 44819195 IC50 > 6000000 nM T06093 C28LAX 44819196 IC50 = 3200000 nM T06093 CJN1M8 44819197 IC50 > 6000000 nM T06093 CPD13F 44819369 IC50 > 6000000 nM T06093 C45VLQ 44819370 IC50 > 6400 nM T06093 CQP26L 44819371 IC50 = 45 nM T06093 C6GRN9 44819372 IC50 = 14 nM T06093 CXPM95 44819373 IC50 = 180 nM T06093 CZ9N8G 44819374 IC50 = 290 nM T06093 CSI0U1 44819541 IC50 = 4 nM T06093 CM3GX4 45102613 IC50 = 781 nM T06093 CA4XQ3 45375859 IC50 = 0.9 nM T06093 CHI0X2 45380476 IC50 < 1 nM T06093 CT6LS4 45380564 IC50 = 8.5 nM T06093 CUGW46 45380655 IC50 < 1 nM T06093 CVXU61 45381162 IC50 = 17.99 nM T06093 C0FM5X 45381385 IC50 = 6565 nM T06093 C7J0OL 45381386 IC50 = 5421 nM T06093 CR2IJ9 45381939 IC50 < 1 nM T06093 C93OTW 46182713 IC50 = 7.8 nM T06093 CYP5E8 46183898 Ki = 2.2 nM T06093 C1MB8Y 46183900 Ki = 0.8 nM T06093 CR0J2W 46184600 Ki = 1 nM T06093 CL3T2P 46184852 Ki = 1.5 nM T06093 COJ06D 46207055 IC50 = 27 nM T06093 CA7Y9E 46207072 IC50 = 67 nM T06093 CNJW82 46207422 IC50 = 3 nM T06093 C9LU8O 46216813 IC50 = 78 nM T06093 CY3HW5 46224684 IC50 = 440 nM T06093 C9XUZ7 46229921 IC50 = 2500 nM T06093 C05RZO 46229922 IC50 > 100000 nM T06093 CZ20AP 46230023 IC50 = 2400 nM T06093 CG3Y2V 46230024 IC50 = 1700 nM T06093 CF7J5W 46230025 IC50 = 6700 nM T06093 CRK5G7 46230026 IC50 = 3000 nM T06093 CO2SM4 46230027 IC50 = 52000 nM T06093 CG0T3I 46230078 IC50 = 45000 nM T06093 C6BVX1 46230079 IC50 = 330 nM T06093 C1W7IZ 46230080 IC50 = 560 nM T06093 C1SVR9 46230081 IC50 = 39 nM T06093 CI5CP4 46230131 IC50 = 62 nM T06093 CAI1J3 46230132 IC50 = 62 nM T06093 CJH61I 46230133 IC50 = 250 nM T06093 C9N5GS 46230134 IC50 = 28 nM T06093 CC09NO 46230135 IC50 = 49 nM T06093 COQ5I4 46230172 IC50 = 21 nM T06093 CEF6C8 46230173 IC50 = 17 nM T06093 CVZ2F7 46230174 IC50 = 89 nM T06093 CDZ1V3 46230175 IC50 = 300 nM T06093 C5UN8M 46230297 IC50 = 5000 nM T06093 C2O0PN 46230298 IC50 = 1200 nM T06093 C5J9UO 46230299 IC50 = 5500 nM T06093 CJUO52 46230300 IC50 = 3500 nM T06093 C2IWB4 46871821 IC50 = 11 nM T06093 CLS29B 46872626 IC50 > 10000 nM T06093 CC5I9X 46879638 IC50 = 9 nM T06093 CDC6H3 46879639 IC50 = 42 nM T06093 C82TLA 46879640 IC50 = 1200 nM T06093 C93DKU 46879641 IC50 = 11 nM T06093 CRW3V8 46879642 IC50 = 25 nM T06093 CE65YR 46879678 IC50 = 47 nM T06093 C69GZJ 46879679 IC50 = 14 nM T06093 CYEB73 46879680 IC50 = 1241 nM T06093 C7H1JY 46879681 IC50 = 314 nM T06093 CF5L9G 46879682 IC50 = 500 nM T06093 C9ZXE5 46879720 IC50 = 66 nM T06093 C0F9PH 46879721 IC50 = 365 nM T06093 CQ29LV 46879722 IC50 = 45 nM T06093 CD5T7Q 46879723 IC50 = 93 nM T06093 C8SEY4 46879724 IC50 = 75 nM T06093 CTB20Y 46879760 IC50 = 1485 nM T06093 CC6AS4 46879761 IC50 = 59 nM T06093 CP9H0C 46879762 IC50 = 7 nM T06093 CGH2F4 46879763 IC50 = 53 nM T06093 CX9O3U 46879803 IC50 = 18 nM T06093 C3Z1KF 46879804 IC50 = 72 nM T06093 CQ5GP8 46879805 IC50 = 59 nM T06093 CQIC19 46879806 IC50 = 26 nM T06093 CCXV26 46879807 IC50 = 94 nM T06093 CISY62 46879865 IC50 = 871 nM T06093 CO16JL 46882137 IC50 = 2.754 nM T06093 C2O8RZ 46886323 IC50 > 1000 nM T06093 C37EBK 46890033 IC50 > 10000 nM T06093 C21PWE 46890034 IC50 = 280 nM T06093 C4XYI7 46890035 IC50 = 430 nM T06093 CXUO70 46890036 IC50 = 26 nM T06093 CJYE86 46890047 IC50 = 8 nM T06093 C5J3HS 46890048 IC50 = 14 nM T06093 C2LZH3 46890049 IC50 = 8 nM T06093 C19RIE 46890050 IC50 = 26 nM T06093 CI3H7X 46890051 IC50 = 9 nM T06093 CO82FC 46890091 IC50 = 210 nM T06093 CNEL95 46890096 IC50 = 4 nM T06093 CX1M2R 46890097 IC50 = 6 nM T06093 CZ2V8R 46890138 IC50 = 110 nM T06093 C54PJN 46890568 IC50 = 31 nM T06093 C15JFA 46890604 IC50 > 10000 nM T06093 CM0QF5 46890605 IC50 > 10000 nM T06093 CAY1H5 46890607 IC50 = 67 nM T06093 CH7OR1 46890608 IC50 = 47 nM T06093 C59PJX 46890609 IC50 = 230 nM T06093 C42PBE 46890610 IC50 = 240 nM T06093 CD31PZ 46890611 IC50 = 6 nM T06093 C3HAB5 46890642 IC50 = 1700 nM T06093 CC3Z1J 46890643 IC50 > 10000 nM T06093 CA3G4C 46890649 IC50 = 6 nM T06093 C0OHA9 46890650 IC50 = 2 nM T06093 CL5NQ1 46890651 IC50 = 4 nM T06093 CG8JF4 46890652 IC50 = 5 nM T06093 CH68YA 46890653 IC50 = 4 nM T06093 CJD2G3 46890690 IC50 > 10000 nM T06093 C9LP4B 46890691 IC50 > 10000 nM T06093 C3MFR6 46890692 IC50 > 10000 nM T06093 C68WFR 46890693 IC50 = 360 nM T06093 CQR9H4 46890702 IC50 = 6 nM T06093 CXQ74C 46890703 IC50 = 11 nM T06093 C85CTL 46890704 IC50 = 7 nM T06093 C8BZF7 46890705 IC50 = 4 nM T06093 C0X7DL 46900277 IC50 = 713 nM T06093 CWK3H1 46900279 IC50 = 18 nM T06093 CW85NG 46900281 IC50 = 1 nM T06093 C13TXR 46900283 IC50 = 22 nM T06093 C9F7WL 46900285 IC50 = 371 nM T06093 CHNB46 46900440 IC50 = 7 nM T06093 CYH8F9 46900589 IC50 = 23 nM T06093 C2G3LX 46900593 IC50 = 156 nM T06093 C78PUX 46900595 IC50 = 850 nM T06093 C2RY0F 46900760 IC50 = 261 nM T06093 CA7PD0 46900762 IC50 = 334 nM T06093 CIVT03 46900765 IC50 = 6 nM T06093 CV1G0H 46900939 IC50 = 25 nM T06093 C8EDL6 46901105 IC50 = 250 nM T06093 CYB7A4 46901107 IC50 = 3 nM T06093 C3SP2O 46901109 IC50 = 190 nM T06093 C2PS4R 46901112 IC50 = 18 nM T06093 CA2Y8J 46901260 IC50 = 2 nM T06093 C96PFW 46901262 IC50 = 18 nM T06093 CXI1R6 46901264 IC50 = 775 nM T06093 CSV5B9 46901859 IC50 = 26 nM T06093 C6E1YT 46938262 Ki = 1.8 nM T06093 CI7C2B 46947635 IC50 < 1 nM T06093 CEPD73 49786965 IC50 = 15 nM T06093 CHSF07 49806372 IC50 > 1000 nM T06093 C1H2PX 49820218 Ki = 6.8 nM T06093 CXG37L 49864747 IC50 = 19 nM T06093 C6LYB5 49864748 IC50 = 20 nM T06093 CE4ZA8 49864749 IC50 = 400 nM T06093 C0XI5Q 49864750 IC50 = 25 nM T06093 C2IM0F 49864793 IC50 = 180 nM T06093 CL6D7S 49864854 IC50 = 310 nM T06093 CA8X0L 49864855 IC50 = 7.3 nM T06093 C6BJ5E 49864856 IC50 = 1000 nM T06093 C5A9SZ 49865528 IC50 = 12 nM T06093 CR38QL 49865529 IC50 = 240 nM T06093 CWTY56 49865530 IC50 = 340 nM T06093 CCL6T7 49870878 IC50 = 575.44 nM T06093 CX6PZ9 51003130 IC50 = 1 nM T06093 CAZQ43 51003133 IC50 > 1000 nM T06093 CDU4Q5 51346827 Ki = 19 nM T06093 C8CGM9 51346966 IC50 > 20000 nM T06093 CXA03W 52920796 IC50 > 100 nM T06093 CC41YU 52933429 IC50 < 1 nM T06093 COGV85 52933915 IC50 = 11 nM T06093 CB24WM 52933916 IC50 < 1 nM T06093 CEW2N3 52933917 IC50 = 3 nM T06093 C4D6ZP 52934146 IC50 = 5 nM T06093 CY8B9U 52934379 IC50 < 1 nM T06093 CD2S0G 52934380 IC50 = 4400 nM T06093 C2Q3AE 52934381 IC50 = 8 nM T06093 C6OA7K 52934832 IC50 = 36 nM T06093 CRDM19 52934834 IC50 = 2300 nM T06093 CU6W0S 52935059 IC50 = 1 nM T06093 CN5Y4M 52935061 IC50 = 160 nM T06093 C5C2HR 52935064 IC50 = 180 nM T06093 C2BTX1 52935500 IC50 = 2 nM T06093 C5UOY3 52935712 IC50 = 24 nM T06093 CF54OU 52935714 IC50 = 310 nM T06093 CAN96R 52935715 IC50 < 1 nM T06093 C9OW2P 52935716 IC50 = 2 nM T06093 C0QF2H 52935717 IC50 = 9 nM T06093 C8IXZ0 52935926 IC50 < 1 nM T06093 C6SW7E 52936149 IC50 = 5 nM T06093 CWV3F9 52936150 IC50 = 220 nM T06093 CEQN27 52936621 Ki > 1000 nM T06093 C6OTY5 53251320 IC50 > 20000 nM T06093 CUQR13 53317664 IC50 = 6 nM T06093 CE8OY2 53317913 IC50 > 100 nM T06093 CCK9X6 53318621 IC50 = 358 nM T06093 C5HD4U 53318622 IC50 > 5000 nM T06093 CZS8K4 53319042 Ki = 44 nM T06093 CYL3C6 53319935 IC50 = 22 nM T06093 CUD21V 53320263 Ki = 62 nM T06093 CRI2V5 53320582 IC50 = 79.43 nM T06093 CV87RK 53321580 IC50 = 3 nM T06093 CRY96M 53321650 IC50 = 1288.25 nM T06093 CESA85 53323614 Ki = 100 nM T06093 C2W9OA 53324451 IC50 > 10000 nM T06093 CUB80V 53325184 IC50 = 6 nM T06093 C9FV6Q 53379585 IC50 = 2.9 nM T06093 C1KYG9 53379691 IC50 = 102 nM T06093 C8NA4L 53384644 IC50 > 30000 nM T06093 CNOA83 53492329 IC50 = 50 nM T06093 C8WFA5 53492330 IC50 = 11 nM T06093 C1XS2J 54760383 IC50 > 10000 nM T06093 CUJM81 54765020 IC50 = 9 nM T06093 CQ28VE 54765021 IC50 = 8 nM T06093 CE0Y9O 54765203 IC50 = 2 nM T06093 C9V7LP 54765280 IC50 = 1 nM T06093 CG7F2E 56603818 IC50 = 9 nM T06093 C04QGT 57390719 IC50 = 200 nM T06093 CR2ZM0 57391854 IC50 = 132 nM T06093 C2UZC6 57392519 IC50 = 2 nM T06093 CJ7HZ1 57392522 IC50 = 3 nM T06093 CJ1EI5 57392627 IC50 = 420 nM T06093 C5RTO0 57394242 IC50 = 43 nM T06093 CJED53 57394243 IC50 = 18 nM T06093 CV4PQ1 57394244 IC50 = 750 nM T06093 C4QK5J 57394245 IC50 = 170 nM T06093 C2OD1C 57394246 IC50 = 290 nM T06093 CAV49N 57394247 IC50 = 18 nM T06093 C5GYP7 57394348 IC50 = 190 nM T06093 CB6U0W 57395100 IC50 = 2 nM T06093 CYU92T 57395101 IC50 < 1 nM T06093 C8BKO6 57395998 IC50 = 9 nM T06093 C3WBE7 57395999 IC50 = 8 nM T06093 C70JBE 57396000 IC50 < 1 nM T06093 C6C7EN 57396001 IC50 = 130 nM T06093 CNH69U 57396872 IC50 = 19 nM T06093 CX24JF 57397800 IC50 = 150 nM T06093 C8R7HP 57397801 IC50 = 4 nM T06093 CBG3T9 57397802 IC50 = 740 nM T06093 C07YVE 57397803 IC50 = 5 nM T06093 CF89DG 57398808 IC50 = 166 nM T06093 C4DM3N 57398809 IC50 = 90 nM T06093 CWG07J 57399140 IC50 < 10 nM T06093 CV6X1C 57399460 IC50 = 3 nM T06093 CH84ZK 57399461 IC50 = 10 nM T06093 C3DR4A 57399462 IC50 = 1900 nM T06093 CG1FJ4 57399463 IC50 = 220 nM T06093 CRA61Q 57399464 IC50 = 220 nM T06093 C6UGL7 57399465 IC50 = 76 nM T06093 C7DT8V 57400298 IC50 = 1 nM T06093 C0JAL7 57400299 IC50 = 6 nM T06093 C0UDY9 57401151 IC50 > 30000 nM T06093 CETA86 57401229 IC50 = 24 nM T06093 CHXD31 57401230 IC50 < 1 nM T06093 CT9NR3 57402100 IC50 < 1 nM T06093 CYUQ67 57402101 IC50 = 1 nM T06093 CL1WN9 57402102 IC50 = 2800 nM T06093 CC41DN 57402103 IC50 = 62 nM T06093 CSEA21 57402104 IC50 = 16 nM T06093 C1F3AS 57402971 IC50 = 7 nM T06093 C8XM3C 57403071 IC50 = 1200 nM T06093 CH5Q0E 57403072 IC50 = 530 nM T06093 CN9G2Z 57403855 IC50 = 8 nM T06093 CTJI57 57404047 IC50 = 1365 nM T06093 CI1A8M 57404048 IC50 = 1608 nM T06093 CPGR16 57404049 IC50 = 247 nM T06093 C2MD4C 57663921 IC50 = 7520 nM T06093 C8X6PU 57663989 IC50 = 5360 nM T06093 C6YAG9 57664030 IC50 = 260 nM T06093 CQP7E0 57750290 IC50 = 39 nM T06093 C1U3YR 57750299 IC50 = 34 nM T06093 CEY8W0 57750311 IC50 = 90 nM T06093 CNBO65 57750312 IC50 = 153 nM T06093 C2F9DS 57750315 IC50 = 351 nM T06093 CZ08KN 57750321 IC50 = 104 nM T06093 CUY8T6 57750329 IC50 = 132 nM T06093 CK4W1L 57750342 IC50 = 112 nM T06093 CM5X9L 57750343 IC50 = 1396 nM T06093 C0TNP8 57750364 IC50 = 182 nM T06093 CBY5E4 57750369 IC50 = 134 nM T06093 CO6P5G 57750381 IC50 = 62 nM T06093 CSI9Y4 57750382 IC50 = 576 nM T06093 C6GH7X 57750391 IC50 = 586 nM T06093 CL7CW0 57750402 IC50 = 204 nM T06093 CA4G5W 57750407 IC50 = 34 nM T06093 CM7XL6 57750408 IC50 = 55 nM T06093 CY4Z8R 57750418 IC50 = 135 nM T06093 C8OY4I 57750420 IC50 = 266 nM T06093 CO7SX4 57920205 IC50 = 40 nM T06093 CBRV34 58310563 IC50 = 9 nM T06093 C81JXL 58310602 IC50 = 1.2 nM T06093 CBGN56 58310712 IC50 = 7 nM T06093 C60ZSA 58897672 IC50 = 540 nM T06093 C6BPR2 58985201 IC50 > 30000 nM T06093 C2NV3R 59198239 IC50 = 10 nM T06093 C86KLG 59563696 Ki = 359 nM T06093 CJ7DQ1 59563724 Ki = 1.7 nM T06093 C6NTI2 59563729 Ki = 4.2 nM T06093 CCS4F7 59563754 Ki = 1 nM T06093 C0VGD1 59563759 Ki = 0.4 nM T06093 CML20P 59563769 Ki = 1.3 nM T06093 C49RWX 59563782 Ki = 0.2 nM T06093 C5IK2H 59563827 Ki = 10.3 nM T06093 CXJ63M 59603829 IC50 = 560 nM T06093 CQEU96 59603842 IC50 = 52 nM T06093 C1MR8Q 60097495 IC50 = 2 nM T06093 CC7A5F 66577033 IC50 < 1 nM T06093 C5F9JE 66906143 Ki = 1.5 nM T06093 C1HSE0 67035086 IC50 = 9 nM T06093 CWI6K5 67035106 IC50 > 10000 nM T06093 CUJ28O 67112053 IC50 > 20000 nM T06093 C2ZJC1 67113434 IC50 > 20000 nM T06093 CK80LJ 67130050 IC50 > 10000 nM T06093 CV63UL 67240318 IC50 > 10000 nM T06093 C90NEZ 67411145 IC50 = 167 nM T06093 C74LIW 67450910 IC50 = 7 nM T06093 C5J8ET 68245749 IC50 = 5.1 nM T06093 C8I7GC 68293638 IC50 > 10000 nM T06093 CD56XK 68293660 IC50 = 6800 nM T06093 CM70FK 68511029 IC50 > 10000 nM T06093 C0UOK4 68512374 IC50 = 96 nM T06093 CLS10P 68513301 IC50 = 1 nM T06093 C5JYB8 68515257 IC50 = 14 nM T06093 CL8SO7 68516150 IC50 = 2400 nM T06093 CKZ4B8 68517263 IC50 = 1 nM T06093 CN0Y5O 68517775 IC50 = 170 nM T06093 C5RPF7 68518614 IC50 > 10000 nM T06093 C78YUA 68518851 IC50 > 10000 nM T06093 CY7DF3 68519300 IC50 = 13 nM T06093 CP8S0Y 68519792 IC50 = 2 nM T06093 C50YAE 68520214 IC50 = 45 nM T06093 CNIM41 68520578 IC50 = 6652 nM T06093 C2VOK4 68521168 IC50 = 7083 nM T06093 CDM0U9 68521184 IC50 = 2358 nM T06093 CM1O5T 68521380 IC50 = 16.98 nM T06093 CAC9S6 68521624 IC50 = 5 nM T06093 C3T6GU 68522253 IC50 = 5570 nM T06093 CE3A0Q 68522320 IC50 = 4508 nM T06093 C8B5YJ 68522434 IC50 = 2572 nM T06093 C4H0PL 68523303 IC50 = 43.95 nM T06093 CHQ9X6 68560451 IC50 = 7.998 nM T06093 C69OHY 68560854 IC50 = 1 nM T06093 C1L8BR 68560881 IC50 = 2 nM T06093 C25MEI 68561431 IC50 = 13 nM T06093 C8ET0B 68561683 IC50 = 33 nM T06093 CP1MZ4 68561726 IC50 = 2 nM T06093 C1E6AQ 68562357 IC50 = 14 nM T06093 C3Z6QH 68562476 IC50 = 2.999 nM T06093 C6XEL5 68562540 IC50 = 1 nM T06093 C8D4TN 68562627 IC50 = 2.999 nM T06093 CXOQ87 68562824 IC50 < 1 nM T06093 C98HZJ 68563012 IC50 > 20000 nM T06093 CCD89X 68563058 IC50 = 1 nM T06093 C02SXB 68563288 IC50 = 2 nM T06093 C7D4GP 68563409 IC50 < 1 nM T06093 CK9PS1 68563527 IC50 = 26 nM T06093 CE0G9W 68563753 IC50 = 751 nM T06093 CFQ95X 68563884 IC50 < 1 nM T06093 C87MSX 68563892 IC50 = 5 nM T06093 CO5DH4 68564018 IC50 = 2.999 nM T06093 CT02PG 68564802 IC50 < 1 nM T06093 C4U2ZW 68565003 IC50 = 12 nM T06093 C0XCY9 68565200 IC50 = 5 nM T06093 CELF91 68565470 IC50 = 2.999 nM T06093 CLF40S 68565711 IC50 = 7 nM T06093 CD94BR 68565840 IC50 = 16.98 nM T06093 CVF0D9 68566096 IC50 < 1 nM T06093 CE71GF 68566105 IC50 = 5.998 nM T06093 CW6BH7 68566254 IC50 = 2 nM T06093 C1GL6M 68566289 IC50 = 611 nM T06093 C2MQ7L 68566290 IC50 = 2 nM T06093 C0HYV6 68566291 IC50 = 1 nM T06093 CP2HY8 68566333 IC50 = 2747.89 nM T06093 C62MNX 68566340 IC50 = 87 nM T06093 CG7T9J 68566450 IC50 = 2 nM T06093 CGQI13 68566531 IC50 < 1 nM T06093 C8Z9FK 68567421 IC50 = 55 nM T06093 CQRP72 68567556 IC50 = 2.999 nM T06093 C3VLM1 68567893 IC50 = 3.999 nM T06093 C48EIQ 68568011 IC50 = 1 nM T06093 CAWC35 68621678 IC50 = 2.5 nM T06093 CA7B3V 68623896 IC50 = 27 nM T06093 C7GRV2 68755406 IC50 > 10000 nM T06093 C5DGR9 69036886 IC50 = 10000 nM T06093 CN7WU6 70681396 IC50 = 32920 nM T06093 CHV21E 70681466 IC50 = 16218.1 nM T06093 C4FD5I 70681467 IC50 < 31622.78 nM T06093 CB95AF 70683491 IC50 = 36100 nM T06093 CGC72H 70683492 IC50 = 19800 nM T06093 C1JT3B 70683589 IC50 < 31622.78 nM T06093 C56GSR 70687744 IC50 > 400000 nM T06093 C6W5DG 70687789 IC50 = 17.78 nM T06093 C5D1LV 70687790 IC50 = 630.96 nM T06093 CW4A2M 70687791 IC50 = 10.23 nM T06093 C8BJC4 70689793 IC50 = 2300 nM T06093 C0GY4P 70689794 IC50 = 1500 nM T06093 CP7N4B 70689795 IC50 = 1070 nM T06093 CVZ96I 70691888 IC50 = 221400 nM T06093 C5YIS3 70691933 IC50 > 400000 nM T06093 C6JEY5 70691934 IC50 = 800 nM T06093 C15BRD 70691935 IC50 = 1100 nM T06093 CZLC64 70691985 IC50 = 151.36 nM T06093 C5V6IR 70693983 IC50 = 7500 nM T06093 CF3H0Y 70694077 IC50 < 31622.78 nM T06093 C93DRT 70696151 IC50 = 34.67 nM T06093 CX7T4B 70696202 IC50 < 31622.78 nM T06093 CM6I3J 70696203 IC50 < 31622.78 nM T06093 CYP62K 70833120 Ki = 0.9 nM T06093 C2TIU0 70833218 Ki = 0.6 nM T06093 C9N8ZJ 70889439 IC50 = 159 nM T06093 C3KRY2 70889465 IC50 = 627 nM T06093 CK9J6L 70896884 IC50 = 24 nM T06093 CNK8P9 70896888 IC50 < 1 nM T06093 CDL35S 70896923 IC50 = 3.999 nM T06093 CF6G7X 71115342 IC50 = 5 nM T06093 C8LM3D 71115401 IC50 < 1 nM T06093 CSJX51 71115438 IC50 = 3.6 nM T06093 CV49YZ 71115454 IC50 = 20 nM T06093 CT0SY1 71115472 IC50 = 4.9 nM T06093 CZJ95T 71115480 IC50 = 5.5 nM T06093 C4UDL5 71115506 IC50 = 1.4 nM T06093 C1WEU9 71115627 IC50 = 48 nM T06093 CMJ5L6 71115650 IC50 = 22 nM T06093 C8GJ1I 71127248 IC50 = 8.7 nM T06093 CBO2D8 71134750 IC50 = 13 nM T06093 CNE41D 71134751 IC50 = 4.3 nM T06093 C9Q6XS 71134754 IC50 = 12 nM T06093 CQ9K7T 71134755 IC50 = 2.7 nM T06093 C64TSZ 71135746 IC50 = 1.4 nM T06093 CV3DN9 71135748 IC50 = 37 nM T06093 C7YBR1 71140511 IC50 = 49 nM T06093 C23NTC 71282961 IC50 < 1 nM T06093 CFPJ95 71283262 IC50 < 1 nM T06093 CT92OL 71295837 IC50 > 10000 nM T06093 CKT60L 71455860 Ki = 430 nM T06093 C89UAF 71505694 IC50 = 2.6 nM T06093 C6WFU1 71505859 IC50 = 1.6 nM T06093 C5TZY7 71505860 IC50 = 2.1 nM T06093 CBHU71 71506022 IC50 < 1 nM T06093 CP68AR 71506023 IC50 < 1 nM T06093 C4AP9J 71506045 IC50 < 1 nM T06093 CE8YU3 71506047 IC50 < 1 nM T06093 CJ5X3M 71506048 IC50 < 1 nM T06093 CC72MW 71506239 IC50 < 1 nM T06093 CAI23O 71506241 IC50 < 1 nM T06093 C2IUD7 71506423 IC50 = 1.3 nM T06093 CZ5AO3 71506424 IC50 < 1 nM T06093 C7PSK9 71506426 IC50 < 1 nM T06093 CARD51 71506616 IC50 < 1 nM T06093 CVZW12 71529762 IC50 = 1.1 nM T06093 CD50QU 71568134 IC50 = 71 nM T06093 C3VH5L 71568135 IC50 = 371 nM T06093 CQV96E 71583048 IC50 = 1297 nM T06093 CSPR52 71583049 IC50 = 3149 nM T06093 CNT5F3 71583050 IC50 = 1144 nM T06093 CH7I0W 71583051 IC50 = 1072 nM T06093 CMY9K6 71607726 IC50 = 1.1 nM T06093 CAZ0M9 71651215 IC50 < 1 nM T06093 C4DUS3 71654759 IC50 = 304 nM T06093 CWC30G 71654760 IC50 = 88 nM T06093 CTR8D3 71654761 IC50 = 1016.25 nM T06093 C03PGX 71654826 IC50 = 279.9 nM T06093 C1XJV9 71654827 IC50 = 253 nM T06093 C8TB9J 71654828 IC50 = 331 nM T06093 CF1O4J 71654829 IC50 = 570 nM T06093 C2FZ7P 71654892 IC50 = 924 nM T06093 C27GJP 71654893 IC50 = 425 nM T06093 C2GKS8 71654894 IC50 = 281 nM T06093 CD32RE 71654895 IC50 = 357 nM T06093 CX8D4B 71654972 IC50 = 2984 nM T06093 C7BMQ0 71654973 IC50 = 3324 nM T06093 C8AM1K 71655603 IC50 = 1 nM T06093 CZ5V1W 72546278 IC50 = 7.8 nM T06093 C0RV6L 72546279 IC50 = 6.2 nM T06093 C5PLI8 72546521 IC50 = 45 nM T06093 C6N4JU 72546522 IC50 = 1.5 nM T06093 CWZ92C 72547020 IC50 = 55 nM T06093 C0DL3F 72698602 IC50 = 0.45 nM T06093 CTK3L4 77461132 EC50 = 260 nM T06093 C7U4DH 77461136 IC50 = 65 nM T06093 CL6C4U 77461137 EC50 = 380 nM T06093 CSV23A 78673872 IC50 = 23 nM T06093 CLOZ06 81689703 IC50 < 1 nM T06093 C5S7CW 86072887 IC50 = 1800 nM T06093 CTW6L4 86072888 IC50 = 720 nM T06093 C0OCM7 86072889 IC50 = 380 nM T06093 CJB2D6 86072906 IC50 = 1700 nM T06093 C5CD0N 86072920 IC50 > 10000 nM T06093 C76IMA 86270887 Ki = 0.4 nM T06093 C0CWM6 86566735 IC50 = 0.18 nM T06093 CC8I0M 86707711 IC50 = 43 nM T06093 C2M9TQ 86764444 IC50 = 0.51 nM T06093 C91YAJ 87405083 IC50 = 2000 nM T06093 CV86ES 87405158 IC50 = 60 nM T06093 CJ64UO 87405222 IC50 = 290 nM T06093 CVXE69 87405226 IC50 = 2500 nM T06093 CSZ1R0 87405236 IC50 = 120 nM T06093 CIMK73 87405291 IC50 = 20 nM T06093 C5GVJ2 87405534 IC50 = 120 nM T06093 CBF43A 87405559 IC50 = 1900 nM T06093 C3JLM0 87405570 IC50 = 30 nM T06093 CB2H3J 87405750 IC50 = 1100 nM T06093 CN78XC 87405776 IC50 = 70 nM T06093 C9MGP8 87405780 IC50 = 190 nM T06093 CV49YW 87405796 IC50 = 680 nM T06093 CF87VX 87405826 IC50 = 240 nM T06093 CK8BI1 87405909 IC50 = 22000 nM T06093 CGX1F3 87405928 IC50 = 110 nM T06093 CX6L9J 87405953 IC50 = 140 nM T06093 C1NCJ9 87405962 IC50 = 15 nM T06093 C5VFE9 87405965 IC50 = 280 nM T06093 C1HMK3 87406217 IC50 = 12000 nM T06093 C34SGC 87406334 IC50 = 50 nM T06093 CX79WB 87406347 IC50 = 42 nM T06093 CSY87D 87406371 IC50 = 30 nM T06093 C20FIU 87406393 IC50 = 2100 nM T06093 CLK39G 87406409 IC50 = 12 nM T06093 C2XI8F 87406410 IC50 = 10 nM T06093 CD4FH9 87406443 IC50 = 120 nM T06093 CKH3D4 87406530 IC50 = 30 nM T06093 C23ORM 87406786 IC50 = 470 nM T06093 CL1TA4 87407566 IC50 = 31100 nM T06093 C74KNV 87408321 IC50 = 130 nM T06093 CK9VP5 87408525 IC50 = 100 nM T06093 CB5A1I 87481281 IC50 = 140 nM T06093 CB5MP3 87482409 IC50 = 2290 nM T06093 CP26RT 88898804 IC50 = 2700 nM T06093 CG1L7F 88898863 IC50 = 3440 nM T06093 C20UYR 89421099 IC50 = 42 nM T06093 CBY10R 89421243 IC50 = 9300 nM T06093 C45QFT 89421265 IC50 = 6300 nM T06093 CM69ZB 89421450 IC50 = 47 nM T06093 C9SB8C 89421561 IC50 = 78 nM T06093 CK4M3W 89424114 IC50 = 180 nM T06093 C1HW4B 89735655 IC50 = 1100 nM T06093 CXT1G5 90654805 IC50 = 76 nM T06093 C8BCJ5 90654806 IC50 = 68 nM T06093 C14UGJ 90654807 EC50 = 760 nM T06093 COA09T 90668074 IC50 = 7 nM T06093 CEN9Z0 90668075 IC50 < 1 nM T06093 C9JW0N 90668076 IC50 = 30 nM T06093 COX43L 90668077 IC50 < 1 nM T06093 CL56TZ 90668078 IC50 = 14 nM T06093 C7Z6AG 90668079 IC50 < 1 nM T06093 CM4P7O 90668080 IC50 = 34 nM T06093 CIT61M 90668081 IC50 < 1 nM T06093 CAIK61 90668082 IC50 = 35 nM T06093 CN67RP 91758287 IC50 = 14 nM T06093 C86EYJ 91806730 Ki = 3.3 nM T06093 C0Y8ZK 91933875 IC50 > 1000 nM T06093 C1E6PA 91938057 IC50 > 1000 nM T06093 CAU45T 91971978 IC50 > 20000 nM T06093 C9R3XZ 102532131 IC50 = 3339 nM T06093 CCRI64 102532132 IC50 > 20000 nM T06093 CK4EN8 117078674 IC50 = 7 nM T06093 CC8XM3 117078749 IC50 = 3 nM T06093 CHQV21 117078751 IC50 = 22 nM T06093 C1KLF8 117078758 IC50 = 24 nM T06093 C7ZL3Q 118715599 IC50 = 11 nM T06093 C8T0AY 118715600 IC50 = 14 nM T06093 C2J3YZ 118715601 IC50 = 120 nM T06093 CRG06J 118715602 IC50 = 20 nM T06093 C7WS3V 118715603 IC50 = 100 nM T06093 CQM81J 118715604 IC50 = 432 nM T06093 CKTL91 118729133 IC50 = 187.93 nM T06093 CQ1KN0 118729134 IC50 = 87 nM T06093 CGIV97 118729135 IC50 = 751.62 nM T06093 CCSF03 118729136 IC50 = 2985.38 nM T06093 CJ45YF 118729137 IC50 = 3324 nM T06093 COP70Z 118729138 IC50 < 1 nM T06093 CGKH02 118729139 IC50 = 170 nM T06093 C24BIT 118732089 IC50 = 976 nM T06093 CTJZ54 118732090 IC50 > 10000 nM T06093 CI38QT 118732092 IC50 = 1605 nM T06093 C1VES6 118732093 IC50 = 1898 nM T06093 CH3ZB0 118732094 IC50 = 3239 nM T06093 CSYA60 118732095 IC50 = 11270 nM T06093 C0K5LC 118732096 IC50 = 4357 nM T06093 C8UN3S 118732097 IC50 > 10000 nM T06093 CW2ZV1 118732098 IC50 = 8940 nM T06093 C4HM7F 118732099 IC50 = 5932 nM T06093 C5QTK1 118732100 IC50 > 10000 nM T06093 C41IOQ 118732101 IC50 = 3219 nM T06093 C2R9JZ 118732102 IC50 > 10000 nM T06093 CZO5W1 118732104 IC50 = 460 nM T06093 C0KG9I 118732105 IC50 > 10000 nM T06093 CR1Z0O 118732106 IC50 > 10000 nM T06093 CYRJ23 118732109 IC50 > 20000 nM T06093 CS7X1V 118737322 IC50 < 1 nM T06093 CWQ05R 118737323 IC50 = 6.6 nM T06093 CPQ46E 118737324 IC50 = 1.5 nM T06093 CI16CF 118737325 IC50 = 3.3 nM T06093 CTB9O6 118737326 IC50 = 1.8 nM T06093 CA0DQ2 118737327 IC50 = 7 nM T06093 C8ZPE0 118737328 IC50 = 27 nM T06093 C9GA8U 118737329 IC50 = 72 nM T06093 CW9UO6 118737330 IC50 = 3.3 nM T06093 CR53GH 118737331 IC50 = 1.8 nM T06093 COW49P 118737332 IC50 < 1 nM T06093 CT7E5V 118737333 IC50 = 1.2 nM T06093 CX9L8M 118737334 IC50 = 1.4 nM T06093 C1P4FO 118737335 IC50 = 2 nM T06093 C0T7PH 118737336 IC50 < 1 nM T06093 CC3MV8 118737337 IC50 = 3.5 nM T06093 CKE9M3 118737373 IC50 < 1 nM T06093 C0CXK9 118737374 IC50 = 1 nM T06093 CG1N5B 118753636 IC50 = 11.2 nM T06093 CQ1TL7 118879520 IC50 = 1330 nM T06093 C68WEZ 121363748 IC50 = 1.16 nM T06093 C7PBG6 122178347 IC50 = 9920 nM T06093 C1ACJ0 122189152 IC50 < 1 nM T06093 CTOX13 122189153 IC50 = 8.9 nM T06093 CA0NQ6 122189154 IC50 = 100 nM T06093 CXK73S 122189155 IC50 = 63 nM T06093 CUYA85 122189156 IC50 = 7.9 nM T06093 CQS34F 122189157 IC50 = 56 nM T06093 CE13UV 122189158 IC50 = 7.2 nM T06093 C4E8IF 122189159 IC50 = 41 nM T06093 CCT83H 122189160 IC50 = 53 nM T06093 CY23RV 122189161 IC50 = 137 nM T06093 CFJR29 122189162 IC50 = 16 nM T06093 CEX47Y 122189163 IC50 = 1.8 nM T06093 CUB9Q5 122189164 IC50 = 62 nM T06093 C63OQZ 122189165 IC50 = 11 nM T06093 CG51VB 122189166 IC50 > 10000 nM T06093 CH74JB 122189167 IC50 = 67 nM T06093 C0SO5F 122189168 IC50 > 1000 nM T06093 CUML53 122189169 IC50 = 2060 nM T06093 C23PWJ 122189170 IC50 = 416 nM T06093 C4M6BZ 122189171 IC50 > 1000 nM T06093 C5ZO6J 122189172 IC50 > 1000 nM T06093 C36LON 122189173 IC50 = 2.5 nM T06093 C5IDL1 122189174 IC50 = 5.7 nM T06093 CTQ9U7 122189175 IC50 = 652 nM T06093 C31YGS 122189176 IC50 > 1000 nM T06093 CC48FJ 122189177 IC50 > 1000 nM T06093 C9Y0PI 122194166 IC50 > 20000 nM T06093 C0C4EH 122194167 IC50 = 2114 nM T06093 C03GHF 122194168 IC50 = 2011 nM T06093 CT56LG 122194169 IC50 = 1021 nM T06093 CJ6AU1 123155509 Ki = 2 nM T06093 C7I5LX 124636147 IC50 = 172 nM T06093 CXT9A0 127026636 Ki = 5.5 nM T06093 C73ZQL 127026938 Ki = 1.3 nM T06093 CAZ1S5 127027580 Ki = 3.2 nM T06093 CCL26O 127027581 Ki = 21.8 nM T06093 C3PFL9 127027582 Ki = 0.8 nM T06093 C0YO6C 127027883 Ki = 821 nM T06093 CJI46K 127027884 Ki = 275 nM T06093 C5W1FY 127027885 Ki = 4.8 nM T06093 CG61LA 127028205 Ki = 1.6 nM T06093 CXE05A 127028206 Ki = 0.7 nM T06093 C9SXG4 127028820 Ki = 3 nM T06093 CZ8YB1 127028821 Ki = 2.7 nM T06093 CQ7FE8 127028822 Ki = 1.8 nM T06093 C70POI 127028823 Ki = 1 nM T06093 C8ZPI9 127028824 Ki = 0.7 nM T06093 CG7RA1 127029119 Ki = 42 nM T06093 CWY0F3 127030602 Ki = 2 nM T06093 CT4G1B 127030603 Ki = 1 nM T06093 CV2BW0 127030609 Ki = 16 nM T06093 C39CBG 127031223 Ki = 1.2 nM T06093 C14PWL 127031251 Ki = 1.3 nM T06093 CR5FK6 127031252 Ki = 0.9 nM T06093 CR74TL 127031527 Ki = 0.4 nM T06093 CQI0T4 127031535 Ki = 0.8 nM T06093 C4C1JA 127031536 Ki = 1 nM T06093 C9W5HD 127031817 Ki = 1 nM T06093 CCS58W 127031818 Ki = 1 nM T06093 CS5T7U 127031819 Ki = 2 nM T06093 CC1VO7 127047444 IC50 = 370 nM T06093 CAW6X5 127047919 IC50 > 1000 nM T06093 C3ORU9 127052113 IC50 = 936 nM T06093 CO47QJ 133054002 IC50 > 20000 nM T06093 C9NL1A 134475022 IC50 = 3 nM T06093 CU2TB7 134823957 IC50 = 21 nM T06093 CDC38O 134823958 IC50 = 37 nM T06093 CR75LH 135894301 IC50 = 16 nM T06093 CX0S1G 135894302 IC50 = 98 nM T06093 CS8R2K 135894303 IC50 = 6 nM T06093 CB48YK 135894304 IC50 = 20 nM T06093 C50ZRD 135894306 IC50 = 9 nM T06093 C3VNE8 135894315 IC50 = 16 nM T06093 C06IBO 135894321 IC50 = 2 nM T06093 CT67YI 135894328 IC50 < 1 nM T06093 C0EYR3 135894330 IC50 = 2 nM T06093 CLOR20 135894333 IC50 = 188 nM T06093 C6G0ZN 135894342 IC50 = 33 nM T06093 C7NIU2 135894347 IC50 < 1 nM T06093 C7QU3Y 135894349 IC50 = 1 nM T06093 CD4SO0 135894350 IC50 < 1 nM T06093 CI7BH2 135894352 IC50 < 1 nM T06093 C75TYJ 135894358 IC50 = 4 nM T06093 C7GR4U 135894359 IC50 = 13 nM T06093 CM2UH4 135894362 IC50 = 9 nM T06093 CT6XZ8 135894363 IC50 = 10 nM T06093 CY19DW 135894364 IC50 = 43 nM T06093 CAF02Z 136030606 IC50 = 18 nM T06093 COT91K 136030607 IC50 = 21 nM T06093 C51OCI 136030637 IC50 > 5000 nM T06093 C0GNY5 136030683 IC50 = 2 nM T06093 C7CB0D 136030684 IC50 < 1 nM T06093 C70WVA 136030685 IC50 = 11 nM T06093 CBK1T7 136030688 IC50 = 123 nM T06093 CPQ9C6 136030689 IC50 = 2 nM T06093 C6PV8U 136030749 IC50 = 423 nM T06093 C7J0VF 136030750 IC50 = 104 nM T06093 C1J0YD 136044172 IC50 < 1 nM T06093 C6HKZ7 136086838 IC50 = 2900 nM T06093 C9ASI3 136086839 IC50 > 10000 nM T06093 CDU3R4 136086840 IC50 > 10000 nM T06093 CVJ42A 136086841 IC50 > 10000 nM T06093 C9X8FI 136141555 IC50 = 31 nM T06093 CPMS45 136141556 IC50 = 87 nM T06093 CH12KM 136141557 IC50 = 3 nM T06093 CVSF01 136188829 IC50 = 6 nM T06093 CDGW87 136188830 IC50 = 1 nM T06093 CLT3N8 136188831 IC50 = 5 nM T06093 CFR6A9 136188832 IC50 = 1 nM T06093 C15HQK 136218656 IC50 = 6 nM T06093 CZ06UK 136218660 IC50 = 1 nM T06093 CML48X 136218661 IC50 < 1 nM T06093 COB69I 136218662 IC50 < 1 nM T06093 CSL6Q8 136218663 IC50 = 5 nM T06093 C6IQF5 136226212 IC50 = 2 nM T06093 CTFJ83 136226213 IC50 = 7 nM T06093 C2SI6E 136226214 IC50 = 19 nM T06093 C2IN8G 136226215 IC50 = 39 nM T06093 C1WT2I 136240901 IC50 = 4 nM T06093 C5EV8A 136240902 IC50 = 13 nM T06093 CX9LB5 136240903 IC50 = 8 nM T06093 C7NJW0 136240904 IC50 = 49 nM T06093 CHWI71 136240905 IC50 = 23 nM T06093 CMC58H 136240944 IC50 = 18 nM T06093 COB58E 136240945 IC50 = 14 nM T06093 CMCH32 136240946 IC50 = 10 nM T06093 C8DET4 136240978 IC50 = 8 nM T06093 CI3KJ1 136241011 IC50 = 225 nM T06093 C60PRZ 136241012 IC50 = 4 nM T06093 CSRD17 136241013 IC50 = 7 nM T06093 CE6X3K 136241014 IC50 = 12 nM T06093 CKQG48 136252254 IC50 = 6 nM T06093 CWB21X 136252255 IC50 = 52 nM T06093 C9MW4C 136252256 IC50 = 239 nM T06093 CKUA76 136252257 IC50 = 88 nM T06093 CC4B3D 136252258 IC50 = 2 nM T06093 C1Q9YN 136252259 IC50 = 8 nM T06093 CW8VD9 136252260 IC50 = 7 nM T06093 CP2IU9 137408384 IC50 = 76 nM T06093 C1TY6N 137631658 IC50 = 2700 nM T06093 CO0XI5 137632168 IC50 > 10000 nM T06093 C8U1CL 137632318 IC50 = 7.3 nM T06093 CP20NK 137633749 IC50 = 7400 nM T06093 CI1E8V 137634241 IC50 = 6320 nM T06093 CSDJ03 137634374 IC50 = 94 nM T06093 C7F5LK 137634439 IC50 = 620 nM T06093 CK5LI2 137634643 IC50 = 2200 nM T06093 CP6Q3K 137634870 IC50 = 5700 nM T06093 C6LQ9T 137634871 IC50 = 900 nM T06093 C49ENV 137635659 IC50 = 1600 nM T06093 CGF95R 137636716 IC50 = 320 nM T06093 C0WQ4T 137637877 IC50 = 1200 nM T06093 CXL97Y 137637941 IC50 > 10000 nM T06093 C1KP4O 137638201 IC50 = 270 nM T06093 CUIS85 137638312 IC50 = 110 nM T06093 CG2JO7 137638433 IC50 = 49 nM T06093 C94BQA 137638520 IC50 = 320 nM T06093 CGP48Y 137639114 IC50 = 7800 nM T06093 CXOK62 137639159 IC50 = 160 nM T06093 CS05VB 137639624 IC50 = 74 nM T06093 C8S9CP 137639731 IC50 > 10000 nM T06093 C3S2CY 137639895 IC50 = 120 nM T06093 CI0O4Z 137640915 IC50 = 190 nM T06093 C1SB6C 137642843 IC50 = 7100 nM T06093 C4MQ5Y 137642906 IC50 = 550 nM T06093 CPJ26N 137642976 IC50 > 10000 nM T06093 CG7Y0B 137644025 IC50 = 2300 nM T06093 CS0YG3 137644558 IC50 = 140 nM T06093 CTF39Y 137644968 IC50 = 260 nM T06093 CVK87P 137645302 IC50 = 350 nM T06093 CV3XS8 137646260 IC50 = 58 nM T06093 C4GH0S 137646432 IC50 = 160 nM T06093 CWQ9E3 137647073 IC50 = 70 nM T06093 C2P6BA 137647099 IC50 > 10000 nM T06093 CX5IK9 137647205 IC50 = 390 nM T06093 C42QMT 137647256 IC50 = 5100 nM T06093 CX5BK1 137647477 IC50 = 76 nM T06093 CI3F0Q 137647696 IC50 = 27 nM T06093 CJF3E2 137648687 IC50 = 6200 nM T06093 C5WL9O 137649838 IC50 = 340 nM T06093 CK2PS3 137649977 IC50 = 31 nM T06093 C0F3WD 137650435 IC50 = 1600 nM T06093 C5OC2K 137650510 IC50 = 50 nM T06093 C1K7RF 137651597 IC50 = 100 nM T06093 CTE9Q3 137652266 IC50 = 1100 nM T06093 CP04RX 137652802 IC50 = 360 nM T06093 CA46UD 137653406 IC50 = 320 nM T06093 C4OB0A 137653917 IC50 = 3200 nM T06093 C7CG5F 137654450 IC50 = 18 nM T06093 C8R0JP 137654554 IC50 = 220 nM T06093 C7NO2X 137654557 IC50 = 85 nM T06093 CQHX89 137654641 IC50 = 98 nM T06093 CGV17I 137654863 IC50 = 530 nM T06093 CF9H2C 137655150 IC50 > 10000 nM T06093 CSW4Y2 137655245 IC50 > 10000 nM T06093 C24DNY 137655381 IC50 = 1400 nM T06093 C4W0VL 137656116 IC50 = 720 nM T06093 CF0PL4 137656779 IC50 = 2600 nM T06093 CR0QK1 137656838 IC50 = 130 nM T06093 CJ9KZ2 137657230 IC50 = 52 nM T06093 CH08TM 137658866 IC50 = 480 nM T06093 C61FIS 137658873 IC50 = 360 nM T06093 C5KX6J 137659805 IC50 = 22 nM T06093 CF42ZX 137660643 IC50 = 540 nM T06093 C9T7CJ 137660696 IC50 = 170 nM T06093 CAPY58 137661040 IC50 = 47 nM T06093 CN6QW0 137661458 IC50 = 1800 nM T06093 CU4BG8 139030519 IC50 = 0.51 nM T06093 CIE59H 139589900 IC50 > 100000 nM T06093 CX7BJ4 139589901 IC50 = 7000 nM T06093 CY9V6D 139589902 IC50 > 100000 nM T06093 C74PTN 139589903 IC50 > 100000 nM T06093 CL06TC 139589904 IC50 = 27000 nM T06093 CE6N7B 139589905 IC50 > 100000 nM T06093 CI6HT9 139589906 IC50 = 42000 nM T06093 C5TR9K 139589907 IC50 = 39000 nM T06093 C2OCB0 139589936 IC50 = 1400 nM T06093 C2W4NJ 139589937 IC50 = 340 nM T06093 CK90DE 139589938 IC50 = 340 nM T06093 C1OXF6 139589939 IC50 = 5.7 nM T06093 C0NCJ7 139589940 IC50 = 910 nM T06093 CNW73T 139589941 IC50 = 40 nM T06093 C1PVA9 139589942 IC50 = 150 nM T06093 CO73YE 139589944 IC50 = 970 nM T06093 CIZ1D6 139590148 IC50 > 20000 nM T06093 C6EK5Y 139590149 IC50 > 20000 nM T06093 CT70MX 139590150 IC50 > 20000 nM T06093 CDNC31 145967951 IC50 > 500 nM T06093 CNXS01 145974852 IC50 = 9000 nM T06093 C5Z6KS 145980871 IC50 = 20 nM T06093 CP97BA 145982455 IC50 = 260 nM T06093 CPL62H 145991717 IC50 = 851 nM T06093 CUC18Q 145992833 IC50 = 29 nM T06093 CNFK73 146585996 IC50 = 547 nM T06093 C14TZG 146586014 IC50 = 1508 nM T06093 CC6W7U 146586023 IC50 = 15 nM T06093 CH30AU 148753963 IC50 = 17 nM T06093 C9UEM2 153496212 IC50 = 62 nM T06093 C8ZPS4 155091368 IC50 = 659.3 nM T06093 CIK53P 155510829 IC50 = 1 nM T06093 CK0X8P 155511505 IC50 = 32 nM T06093 C7ZE5Q 155511547 IC50 = 87 nM T06093 CH3FV7 155512419 IC50 = 41 nM T06093 C2MD1Q 155513187 IC50 = 3 nM T06093 C85BYR 155514878 IC50 = 58 nM T06093 C49AVE 155517210 IC50 = 999 nM T06093 CJR09L 155517677 IC50 = 6894 nM T06093 CW92OR 155517870 IC50 = 84 nM T06093 C7JNV6 155518154 IC50 = 10 nM T06093 CSC9D7 155518157 IC50 = 220 nM T06093 CMAU36 155518545 IC50 = 7 nM T06093 C8VJ0R 155519127 IC50 = 3800 nM T06093 CSNO68 155519979 IC50 = 98 nM T06093 CRE3V4 155521980 IC50 = 5 nM T06093 CX87AL 155522068 IC50 = 49 nM T06093 CRI75C 155522515 IC50 = 374 nM T06093 C1GW0T 155522588 IC50 = 176 nM T06093 C57TCD 155523512 IC50 = 15 nM T06093 C12KNB 155523817 IC50 = 110 nM T06093 CJH7B6 155524106 IC50 = 3526 nM T06093 C5Y7IU 155524764 IC50 = 27 nM T06093 CF0XQ6 155525891 IC50 = 22 nM T06093 C8DC7J 155526399 IC50 = 8 nM T06093 CZ1Y2X 155526562 IC50 = 4163 nM T06093 C5UDL7 155527182 IC50 = 24 nM T06093 CWA7T8 155527595 IC50 = 22 nM T06093 CI31SP 155527821 IC50 = 27 nM T06093 C35MHA 155528108 IC50 = 652 nM T06093 C6KQC9 155529602 IC50 = 34 nM T06093 CFW4G8 155530204 IC50 > 10000 nM T06093 CET2B6 155531372 IC50 = 14 nM T06093 CO7Q5Z 155532093 IC50 = 899 nM T06093 C7F6MP 155532760 IC50 = 15 nM T06093 CS08FU 155533862 IC50 = 15 nM T06093 COLR41 155533909 IC50 = 6 nM T06093 CX86LP 155534718 IC50 = 33 nM T06093 CR6EI1 155535218 IC50 = 3800 nM T06093 C2EJP6 155535544 IC50 = 180 nM T06093 CZ4U1M 155535897 IC50 = 66 nM T06093 COX2T3 155536115 IC50 = 136 nM T06093 C76VOG 155536890 IC50 = 263 nM T06093 CYV7C2 155537163 IC50 = 1283 nM T06093 C8K3XJ 155537606 IC50 = 12 nM T06093 CE8H4O 155537760 IC50 = 9974 nM T06093 C6QM4V 155537815 IC50 = 7102 nM T06093 CL42XY 155537848 IC50 = 83 nM T06093 C6ZB3U 155538076 IC50 = 1300 nM T06093 CJ50ZQ 155538379 IC50 = 9 nM T06093 CDU52V 155538567 IC50 = 118 nM T06093 CO7J3N 155539166 IC50 = 1345 nM T06093 CXP3U1 155539357 IC50 > 10000 nM T06093 CD8N7Z 155541709 IC50 = 43 nM T06093 CLD14S 155542848 IC50 = 82 nM T06093 C1KM6E 155544122 IC50 = 302 nM T06093 C2VC7N 155544946 IC50 = 2027 nM T06093 CNF7U3 155545164 IC50 > 10000 nM T06093 C1R5IF 155546763 IC50 = 29 nM T06093 CHEF57 155549647 IC50 = 306 nM T06093 C8U0DB 155550541 IC50 = 320 nM T06093 CZ5PL2 155552103 IC50 = 14 nM T06093 C2AZ8C 155553393 IC50 = 270 nM T06093 CXB5H9 155553912 IC50 = 140 nM T06093 CPV5G8 155555193 IC50 = 169 nM T06093 C14YJN 155555691 IC50 = 12 nM T06093 C04UNO 155556381 IC50 = 21 nM T06093 C2TMB4 155556732 IC50 = 68 nM T06093 CRP51F 155556776 IC50 = 34 nM T06093 C56FHU 155557272 IC50 = 19 nM T06093 C0QTC9 155557377 IC50 = 77 nM T06093 CNH27R 155557555 IC50 = 700 nM T06093 C64CJZ 155557560 IC50 = 85 nM T06093 CSO32E 155557808 IC50 = 5738 nM T06093 C0C9PZ 155559054 IC50 = 5 nM T06093 C6A4MZ 155560497 IC50 > 10000 nM T06093 CJ1D6M 155560595 IC50 = 2149 nM T06093 CFBY89 155560747 IC50 = 390 nM T06093 CLE6M4 155561562 IC50 = 4557 nM T06093 CK7IN8 155562339 IC50 = 72 nM T06093 CU8W7G 155564298 IC50 = 250 nM T06093 CS19LR 155564577 IC50 > 10000 nM T06093 CWI5K3 155564704 IC50 = 3141 nM T06093 CDU87W 155565976 IC50 = 3 nM T06093 CC1IQ5 155566548 IC50 > 10000 nM T06093 CL1MB0 155567304 IC50 = 75 nM T06093 CSQ69A 155567470 IC50 > 10000 nM T06093 CWMC47 155567479 IC50 = 54 nM T06093 C98WUH 155567548 IC50 = 16 nM T06093 CX91DZ 155567940 IC50 = 350 nM T06093 CT86WS 155568736 IC50 = 4206 nM T06093 D00ERW 44444843 Ki > 7500 nM T06093 D00HVA 11624601 Ki > 7500 nM T06093 D03CPB 60138149 IC50 = 6 nM T06093 D05JRA 25190769 IC50 = 10.47 nM T06093 D06HVH 54613583 IC50 = 220 nM T06093 D07ADX 54764565 IC50 = 111 nM T06093 D07UBK 46911016 IC50 = 100 nM T06093 D07XWC 44477445 IC50 = 2700 nM T06093 D09FFE 449241 IC50 = 3630.78 nM T06093 D0F8HX 12967404 IC50 = 11 nM T06093 D0J7YE 17164245 IC50 = 40000 nM T06093 D0L1UK 3064778 IC50 = 575.44 nM T06093 D0ME9B 46868971 IC50 > 10 nM T06093 D0N1UU 46871820 IC50 = 4 nM T06093 D0Q3NG 11715520 Ki > 7500 nM T06093 D0R3MO 46864283 IC50 < 1 nM T06093 D0S7IE 11658882 Ki > 7500 nM T06093 D0U8UK 11677079 IC50 = 1400 nM T06093 D0V0KA 24863112 IC50 = 19 nM T06093 D0Y5RO 4566 IC50 = 600 nM T31309 D00PBX 49846579 Ki < 0.01 nM T31309 D02OZK 11404337 EC50 = 300 nM T31309 D05TPI 72276 Ki > 100000 nM T31309 D06ETI 24978538 Ki < 0.01 nM T31309 D0I5DP 118910268 Ki = 950 nM T31309 D0Q7AG 53240420 IC50 > 50000 nM T31309 D0U2BH 65064 Ki = 234.42 nM T31309 D0Z0HH 3503 Ki = 170 nM T31309 D03TTE 135513044 Ki = 35 nM T31309 D0B1UL 136002683 Ki = 150 nM T31309 D0CR9A 136183441 Ki = 170 nM T31309 D0L8WH 11228183 Ki < 0.6 nM T31309 CU12QE 1203 Ki > 100000 nM T31309 CK4N7S 6293 Ki = 1150 nM T31309 CQ6B2R 11768 Ki = 583 nM T31309 CX4FN2 65084 Ki > 100000 nM T31309 CG02DS 68258 IC50 = 4300000 nM T31309 CTK25Q 72277 Ki > 100000 nM T31309 C5KW4H 72311 Ki = 171000 nM T31309 CJUW83 95696 Ki > 1000000 nM T31309 CNIW58 107905 Ki = 229.09 nM T31309 C5ZLW6 114777 Ki = 690 nM T31309 C6FK9M 196978 Ki = 1700 nM T31309 CDZ65K 199472 Ki = 235 nM T31309 CY69TA 222032 IC50 = 7700 nM T31309 CBXG18 245869 Ki = 831.76 nM T31309 CP56OU 341016 IC50 = 14000 nM T31309 CBT9L4 434797 IC50 = 5800 nM T31309 C76CAZ 719016 Ki > 1000000 nM T31309 CMP56I 815185 Ki > 1000000 nM T31309 C08YVK 819258 Ki > 1000000 nM T31309 C7GY1X 869152 Ki > 10000 nM T31309 CB7I6E 1549842 Ki > 10000 nM T31309 CRV86S 1555114 Ki = 115000 nM T31309 CJ5TR3 1576659 Ki = 14200 nM T31309 CGAM30 1582605 Ki = 54650 nM T31309 CC74TR 2771353 Ki = 6090 nM T31309 CS5N4Q 3101542 Ki = 3000 nM T31309 CPS79F 3163284 Ki > 1000000 nM T31309 CPCI25 3355449 IC50 = 11700 nM T31309 CRP38E 4369509 IC50 = 93 nM T31309 CLM65T 5276454 Ki = 230 nM T31309 C3IUN5 5720188 Ki = 2400 nM T31309 CR2V0Y 6090108 Ki = 43400 nM T31309 C3JX7W 6484626 Ki > 1000000 nM T31309 C3FIT9 6512895 IC50 = 8000 nM T31309 CVBR15 6520864 IC50 = 3200 nM T31309 COG3E6 6535736 IC50 = 3100 nM T31309 CJU75C 7655492 Ki = 7430 nM T31309 C9UG3Y 10616967 Ki > 50000 nM T31309 CV1X4J 11031986 Ki = 420 nM T31309 CDAT72 11433190 Ki > 10000 nM T31309 C2VTX5 11498270 Ki = 1980 nM T31309 CXK63W 11498475 Ki = 55 nM T31309 C1FO6C 11500877 Ki = 310 nM T31309 CV4JK3 11502754 IC50 > 100000 nM T31309 CVE4N6 11512578 IC50 > 50000 nM T31309 CJI08E 11512941 Ki = 3260 nM T31309 C23QHG 11513027 Ki = 92.1 nM T31309 CU6KI5 11513202 Ki = 366 nM T31309 CQY3D8 11527399 Ki = 721 nM T31309 C8U6YE 11527635 Ki = 110 nM T31309 CH6ZQ5 11541165 Ki > 10000 nM T31309 CKQ0Y7 11542308 Ki = 116 nM T31309 CMZ16P 11556440 Ki = 62 nM T31309 C6EIC4 11585288 Ki = 3540 nM T31309 CATI96 11585498 Ki = 75 nM T31309 C3H1IL 11585607 Ki = 732 nM T31309 CI1U6J 11607072 Ki > 10000 nM T31309 CRY85Q 11607405 Ki = 70 nM T31309 CZCQ84 11614246 Ki = 4570 nM T31309 CNE9T7 11614353 Ki = 1260 nM T31309 CJG0E3 11621908 Ki = 2160 nM T31309 C6HB9W 11643296 Ki = 402 nM T31309 CPX8O4 11649997 Ki > 10000 nM T31309 CJI48S 11650712 Ki = 121 nM T31309 CE3W8S 11657048 Ki = 192 nM T31309 C5SLF8 11657862 Ki = 58.8 nM T31309 C2O6HD 11679126 Ki = 400 nM T31309 CVL56F 11686025 Ki = 231 nM T31309 C0T9EK 11686478 Ki = 165 nM T31309 CJN6Y0 11700195 Ki = 2880 nM T31309 CRIF42 11707282 Ki = 1230 nM T31309 C3PY5U 11707606 Ki = 317 nM T31309 C9U7TI 11721651 Ki = 73 nM T31309 C8TQX1 12158631 Ki = 340 nM T31309 CY56QF 13369486 Ki = 474760 nM T31309 CM7DS2 15991562 Ki = 67 nM T31309 C34ZAH 16072153 Ki = 2850 nM T31309 C7KB3S 16090305 Ki = 930 nM T31309 C9XZU1 16090306 Ki = 25000 nM T31309 C8IBM3 16109062 Ki = 16 nM T31309 CCSZ31 16109063 Ki = 20 nM T31309 C82PXV 16109064 Ki = 8.1 nM T31309 CD95NJ 16109065 Ki = 1.8 nM T31309 CRFU59 16109066 Ki = 3.1 nM T31309 CFQH70 16109067 Ki = 1.6 nM T31309 C07EWL 16109068 Ki < 1 nM T31309 CP1KE4 16109069 Ki < 1 nM T31309 CJ3ND2 16109076 Ki = 3.4 nM T31309 C15FQX 16109077 Ki = 0.7 nM T31309 COB84K 16109078 Ki = 2 nM T31309 C8NB6V 16109079 Ki = 2 nM T31309 C04ZCD 16109080 Ki = 13 nM T31309 CF9P2Y 16109081 Ki = 68 nM T31309 C4XDV1 16109084 Ki = 35.2 nM T31309 C5Q7XJ 16109088 Ki = 6.1 nM T31309 C6NWT1 16109089 Ki = 39.8 nM T31309 CVL8S5 16109090 Ki = 4.5 nM T31309 CUQ1N6 16109091 Ki < 1 nM T31309 CDHV39 16109092 Ki = 3.5 nM T31309 CXV9B1 16109093 Ki < 1 nM T31309 CMU3K7 16109094 Ki < 1 nM T31309 CN9EX7 16109095 Ki = 1 nM T31309 CXD2P4 16109096 Ki < 1 nM T31309 CX0G5D 16109097 Ki = 16.9 nM T31309 CW1R3F 16109098 Ki < 1 nM T31309 C6AX1T 16109099 Ki < 1 nM T31309 CUP40E 16109115 Ki = 9.6 nM T31309 C8TZ0R 16109116 Ki = 61.9 nM T31309 CF32ZY 16109117 Ki = 300 nM T31309 CHF2Y6 16109137 Ki = 56 nM T31309 C45VIE 16109138 Ki = 6.6 nM T31309 CJ65GB 16109139 Ki < 1 nM T31309 C6MKC4 16109140 Ki = 2.7 nM T31309 CT5R1N 16109141 Ki = 1.4 nM T31309 CSJ4A2 16109142 Ki = 1.5 nM T31309 CVS90W 16109149 Ki = 2.5 nM T31309 CT8Z1X 16109150 Ki = 2.1 nM T31309 CZ9OK8 16109151 Ki = 9.4 nM T31309 CD8C4M 16109152 Ki = 46 nM T31309 CR83BQ 16109153 Ki < 1 nM T31309 C5CTU8 16109154 Ki = 6.5 nM T31309 CKH97W 16109156 Ki = 3.2 nM T31309 C5NC8O 16109157 Ki = 4.6 nM T31309 C0QHV3 16109158 Ki < 1 nM T31309 CHP79I 16109159 Ki < 1 nM T31309 C6IZ8J 16109160 Ki < 1 nM T31309 CV8AB2 16109161 Ki < 1 nM T31309 C75YUM 16109162 Ki < 1 nM T31309 CI4Y5D 16109163 Ki < 1 nM T31309 C2Y3HZ 16204196 Ki = 3100 nM T31309 CJV1O2 16204197 Ki = 590 nM T31309 CV7HC8 16645886 Ki > 1000000 nM T31309 CZVP08 16735295 Ki = 17 nM T31309 CO38KM 16735541 Ki = 730 nM T31309 C49JYU 22683787 Ki > 1000000 nM T31309 C5NI1B 24798804 IC50 = 8.7 nM T31309 C9MNJ7 24800647 IC50 = 41600 nM T31309 CNQF59 24800648 IC50 = 3400 nM T31309 CJB1U9 24801007 IC50 = 2600 nM T31309 CN61HR 24801008 IC50 = 290 nM T31309 C07LMB 25059310 Ki = 0.044 nM T31309 C57XNW 25083122 IC50 = 29070 nM T31309 C7GHE9 25099966 Ki > 10000 nM T31309 C4Z7CN 25100119 Ki = 2700 nM T31309 C74OSJ 25100590 Ki > 15000 nM T31309 CHEZ64 25113117 IC50 = 30 nM T31309 C8BO3Z 25117878 Ki < 1 nM T31309 C12LTS 25117879 IC50 = 11 nM T31309 CN5K3H 25117880 Ki < 1 nM T31309 CMF36X 25118047 Ki < 1 nM T31309 C79YVT 25118234 Ki < 1 nM T31309 C3PT2A 25118948 Ki < 1 nM T31309 C2N6XK 25119663 Ki < 1 nM T31309 CHE29K 25138716 Ki < 1 nM T31309 C7F3OP 25138718 Ki = 2.4 nM T31309 CYM3C6 25139034 Ki < 1 nM T31309 C3DPK6 25139036 Ki < 1 nM T31309 C09PGV 25139347 Ki < 1 nM T31309 CCN9B6 25139493 Ki < 1 nM T31309 CN80IZ 25139495 Ki < 1 nM T31309 C1LXT5 25139760 Ki < 1 nM T31309 CT36UD 25140036 Ki < 1 nM T31309 CZU32B 25140188 Ki < 1 nM T31309 CZ9O5H 25140767 Ki < 1 nM T31309 CZQ0K1 25181390 IC50 = 30 nM T31309 C8ULM7 25181391 IC50 = 800 nM T31309 CZ12DX 25229694 Ki = 360 nM T31309 CU34VF 25232834 IC50 = 5000 nM T31309 C6L8MK 25256801 IC50 = 210 nM T31309 C68YHX 26378673 Ki = 320000 nM T31309 C6GOQ2 27433194 Ki = 69600 nM T31309 CK78WE 42601456 Ki = 500 nM T31309 CY9CP3 42613557 Ki = 445 nM T31309 CA9JF3 44191246 IC50 = 4400 nM T31309 C2FXA3 44191638 IC50 = 700 nM T31309 CXO2S9 44191694 IC50 = 150 nM T31309 CHT92S 44191696 IC50 = 670 nM T31309 C83UCJ 44191750 IC50 = 700 nM T31309 CMS39X 44191815 IC50 = 480 nM T31309 C0J3RT 44192144 IC50 = 490 nM T31309 C97RQU 44192145 IC50 = 710 nM T31309 C57VCY 44224066 IC50 = 320 nM T31309 C9LW6U 44224145 IC50 = 42 nM T31309 C5S0YV 44251267 Ki = 1200 nM T31309 CP7O6U 44286285 IC50 ~ 9000 nM T31309 CO5G0M 44357033 IC50 = 3300 nM T31309 C4C7FX 44357034 IC50 = 9000 nM T31309 CDI2R4 44404769 IC50 = 2880 nM T31309 C8LBP2 44404770 IC50 = 1330 nM T31309 C5N2AO 44429172 Ki = 12000 nM T31309 CC5MY2 44429173 Ki = 13500 nM T31309 CO35QT 44429175 Ki = 21200 nM T31309 CR40TC 44429176 Ki = 57800 nM T31309 CDK47L 44429177 Ki = 1950 nM T31309 C4UFY2 44429178 Ki = 192000 nM T31309 CMT5V4 44429179 Ki = 70000 nM T31309 C2XAH8 44429180 Ki > 1000000 nM T31309 CRV49G 44429181 Ki = 260000 nM T31309 C9LM6H 44448452 Ki = 1288.25 nM T31309 CI37EA 44448535 Ki > 100000 nM T31309 CG35DU 44456125 Ki = 260000 nM T31309 CLF8A1 44456175 Ki = 161000 nM T31309 C59ZEM 44456176 Ki = 226000 nM T31309 CAZ5T0 44456210 Ki = 243000 nM T31309 CV43WR 44456211 Ki > 1000000 nM T31309 C85FLZ 44456249 Ki = 21200 nM T31309 C4W6OL 44456329 Ki = 4300 nM T31309 C5MP1Y 44456362 Ki = 4300 nM T31309 CHKW90 44456365 Ki = 1700 nM T31309 CW38KC 44564607 IC50 = 600 nM T31309 CQ4OJ8 44564608 IC50 = 175 nM T31309 C43ZNQ 44564627 IC50 = 1070 nM T31309 C89ODV 44570033 IC50 = 2500 nM T31309 C14DFN 44570035 IC50 = 10700 nM T31309 C7N5RX 44570037 IC50 = 1400 nM T31309 CQVZ10 44570038 IC50 = 190 nM T31309 CV3UF7 44570039 IC50 = 110 nM T31309 CE02OU 44570040 IC50 = 160 nM T31309 C8R1DI 44570041 IC50 = 730 nM T31309 CQ41VK 44570042 IC50 = 1050 nM T31309 CR8FD9 44570043 IC50 = 5610 nM T31309 CNS2K6 44570044 IC50 = 280 nM T31309 C04LUM 44570045 IC50 = 150 nM T31309 C6UFI7 44570046 IC50 = 140 nM T31309 CSND68 44570049 IC50 = 2010 nM T31309 C2DN6W 44570050 IC50 = 100 nM T31309 CJ5L1D 44570051 IC50 = 380 nM T31309 C8DP1H 44570052 IC50 = 650 nM T31309 CW3R7E 44570076 IC50 = 1500 nM T31309 C9M1TK 44570077 IC50 = 50000 nM T31309 CSB46O 44570078 IC50 = 2300 nM T31309 C8RH7P 44570079 IC50 = 3000 nM T31309 CXQ1R9 44570080 IC50 = 1900 nM T31309 CQV64S 44570081 IC50 = 7700 nM T31309 C76VGH 44570082 IC50 = 110 nM T31309 C8S1NW 44570084 IC50 = 210 nM T31309 CDMF54 44570085 IC50 = 50 nM T31309 C3OF5Z 44570086 IC50 = 17300 nM T31309 C43VFD 44570087 IC50 = 20 nM T31309 C25IGP 44570088 IC50 = 90 nM T31309 CK7BQ6 44570089 IC50 = 810 nM T31309 CZB28J 44570090 IC50 = 40 nM T31309 CV78GC 44570091 IC50 = 40 nM T31309 CTFS76 44570092 IC50 = 250 nM T31309 C6TYQ1 44570093 IC50 = 20 nM T31309 C2D1PO 44570094 IC50 = 130 nM T31309 CCF29W 44570095 IC50 = 600 nM T31309 CG0OD4 44570096 IC50 = 510 nM T31309 CH95IX 44574943 Ki = 2000 nM T31309 CFD72X 44574944 Ki = 1300 nM T31309 CNO53W 44574945 Ki = 2500 nM T31309 C5YJF8 44574946 Ki = 1500 nM T31309 CH17BO 44574947 Ki = 3000 nM T31309 CHR74A 44574948 Ki = 1600 nM T31309 C68BOZ 44574949 Ki = 4300 nM T31309 C63BKT 44574950 Ki = 14000 nM T31309 CYD32H 44574951 Ki = 4100 nM T31309 CF6WN0 44574952 Ki = 5400 nM T31309 CNCZ86 44574953 Ki = 7800 nM T31309 CJTI53 44574954 Ki = 8400 nM T31309 CN02TB 44574955 Ki = 2200 nM T31309 CM45OJ 44574956 Ki = 5200 nM T31309 CQ9SA5 44574957 Ki = 6800 nM T31309 CT5F3S 44593461 IC50 = 1100 nM T31309 CH2E4R 44609307 Ki = 8820 nM T31309 CG2NH7 46236925 IC50 = 320 nM T31309 C78NZA 46236926 IC50 = 430 nM T31309 C3DV7L 46701726 Ki = 140 nM T31309 C05NAZ 46836111 Ki = 0.14 nM T31309 CPDE67 46836168 Ki = 150 nM T31309 CF2ZB4 46836243 Ki = 90 nM T31309 CRG96F 46836244 Ki = 100 nM T31309 CY1XE2 46836305 Ki = 240 nM T31309 C8ZHR7 46836862 Ki = 170 nM T31309 CSZT49 46837053 Ki = 220 nM T31309 CL18SN 46887149 IC50 = 11100 nM T31309 C9E3RI 46887150 IC50 = 19400 nM T31309 C3PY8D 49840813 Ki = 1460 nM T31309 C74IAL 49846946 Ki < 0.01 nM T31309 C6HI9D 50899827 Ki = 40 nM T31309 C6TAV4 51002999 Ki = 278 nM T31309 C0J4PO 51003000 Ki = 304 nM T31309 CVBX71 51003001 Ki = 252 nM T31309 CWQ69L 51003061 IC50 = 945 nM T31309 C9USE3 51003064 IC50 = 342 nM T31309 C8BZY6 51003123 IC50 = 302 nM T31309 CQ2X4R 51003124 Ki = 382 nM T31309 C8FYS6 51039416 IC50 = 740 nM T31309 C2ZT6I 51354614 IC50 = 21 nM T31309 C73DOP 51354615 IC50 = 13 nM T31309 CNA1W2 51354616 IC50 = 81 nM T31309 C4Q3YN 51354902 IC50 = 12 nM T31309 CON3Q1 51354903 IC50 = 21 nM T31309 C52OHD 51354904 IC50 = 5 nM T31309 CM3CU0 51355193 IC50 = 84 nM T31309 CJG4D9 52940882 Ki = 5200 nM T31309 CY83NK 52942061 Ki = 5000 nM T31309 C8D2TX 52942120 Ki = 460 nM T31309 C5O2PI 52943275 Ki = 20000 nM T31309 C7I5YW 52944234 Ki = 220 nM T31309 CQTC82 52945653 Ki = 3400 nM T31309 CPA63U 52946674 Ki = 110 nM T31309 CXR6Q3 52946927 Ki = 4600 nM T31309 C1J7UF 52948088 Ki = 12000 nM T31309 C6YCL0 52948158 Ki = 8000 nM T31309 C74FSX 52949135 Ki = 200 nM T31309 CEJT65 52949336 Ki = 83000 nM T31309 CRG5J1 52949401 Ki > 1000 nM T31309 C81RNM 52949424 Ki > 1000 nM T31309 CF5ST9 52950126 Ki = 5800 nM T31309 CW9IN1 53234692 Ki = 1670 nM T31309 CWTA43 53234693 Ki = 1090 nM T31309 CTPX94 53234694 Ki = 1400 nM T31309 CC34HU 53234695 Ki = 930 nM T31309 CHL4C7 53234842 Ki = 760 nM T31309 CZ8TK7 53234845 Ki = 800 nM T31309 CS1ZG8 53235008 Ki = 9490 nM T31309 C6BA1V 53235009 Ki = 3780 nM T31309 CV75RW 53235092 Ki = 3390 nM T31309 C2K5GP 53235093 Ki = 830 nM T31309 C9JD1C 53235169 Ki = 15190 nM T31309 C8KQ6V 54578933 Ki = 158 nM T31309 CRO6I8 54769781 Ki = 1430 nM T31309 CZ1E8X 54769782 Ki = 6031 nM T31309 C7WQI6 54769783 Ki = 886 nM T31309 CO7DE8 54769992 Ki = 16600 nM T31309 CU4RQ6 56933429 IC50 = 2 nM T31309 CNKE09 56933430 IC50 = 1.8 nM T31309 CS3YP8 56933431 Ki < 1 nM T31309 C07IBG 56973535 IC50 = 37 nM T31309 CCN5O6 56973540 IC50 = 190 nM T31309 C9CEO1 57338853 Ki = 179 nM T31309 C38QHP 57339126 Ki = 78000 nM T31309 C5XN9L 57394832 Ki = 3520 nM T31309 CSM8T4 57398377 Ki = 3380 nM T31309 CXP56B 57523339 Ki < 0.6 nM T31309 CX8EG1 57523340 Ki < 0.6 nM T31309 CC3KU7 57523369 Ki < 0.6 nM T31309 COA97D 57523370 Ki = 1.5 nM T31309 C61FYR 57523400 Ki = 8.5 nM T31309 CQ3L5W 57523401 Ki = 21.8 nM T31309 CH3I5T 57523430 IC50 > 100000 nM T31309 C8P2QI 57523431 Ki = 138000 nM T31309 CX9BE7 57523432 IC50 = 0.6 nM T31309 CF6IZ8 57523433 Ki = 1.2 nM T31309 C1YTI4 57523468 Ki = 21.1 nM T31309 C9AFI7 57523469 Ki = 11.6 nM T31309 C0OMZ9 57523470 Ki < 0.6 nM T31309 C4RDZ5 57523498 Ki = 0.8 nM T31309 C5LM1Z 58531411 IC50 = 35 nM T31309 CRN79Z 59053435 IC50 = 19 nM T31309 CHM9V8 59053436 IC50 = 0.9 nM T31309 C6Y1KZ 59053563 IC50 = 110 nM T31309 CNFW46 59053624 IC50 = 5 nM T31309 CJHN01 59053688 IC50 = 140 nM T31309 CL8B3J 59053755 IC50 = 3.8 nM T31309 C40SFQ 59053932 IC50 = 5.6 nM T31309 CS0GE4 59054194 Ki = 4.6 nM T31309 CIR74F 59438327 IC50 > 10000 nM T31309 C04ELI 59447491 Ki = 280 nM T31309 CW1MT4 59447501 Ki = 90 nM T31309 CQF73L 59447527 Ki = 60 nM T31309 CYK9T2 59447570 Ki = 88 nM T31309 CBLR64 59447577 Ki = 74 nM T31309 CN28ME 60169704 Ki < 1 nM T31309 CI13RU 60169705 IC50 = 99 nM T31309 C49HLF 60169795 IC50 = 1.4 nM T31309 C3GRZ0 60204010 Ki < 1 nM T31309 CZPD50 66561644 IC50 = 16 nM T31309 CUVL40 66561645 IC50 = 35 nM T31309 CQ8MS0 66561714 IC50 = 9 nM T31309 CR2Y5X 66561715 IC50 = 15 nM T31309 C0DV3M 66561716 IC50 = 9 nM T31309 C3GH9F 70495544 IC50 = 3.8 nM T31309 CZM1G2 70495760 IC50 = 3.7 nM T31309 CUM37L 70496039 IC50 = 7.1 nM T31309 C2W5BS 70680244 Ki = 870 nM T31309 CF5OC7 70680245 Ki = 5300 nM T31309 C34TMX 70681580 IC50 = 170 nM T31309 CG53LQ 70681581 IC50 = 22 nM T31309 C85SWT 70681582 IC50 = 190 nM T31309 CK5G2S 70681583 IC50 = 120 nM T31309 CT92UD 70681589 IC50 = 180 nM T31309 CGO1Z2 70681590 IC50 = 37 nM T31309 CBWI18 70683696 IC50 = 8 nM T31309 CV01CQ 70683697 IC50 = 71 nM T31309 C5ZGR4 70683707 IC50 = 160 nM T31309 C4R9SX 70683708 IC50 = 14 nM T31309 C1FAS8 70683709 IC50 = 26 nM T31309 CJ3YR9 70684416 Ki = 2 nM T31309 C5QD1R 70685844 IC50 = 140 nM T31309 CR4CN7 70685853 IC50 = 140 nM T31309 CCFR15 70685854 IC50 = 35 nM T31309 CTYS31 70686561 Ki = 15.4 nM T31309 C76YLJ 70687968 IC50 = 4190 nM T31309 CM4L9Q 70687969 IC50 = 45 nM T31309 CL5ZN3 70687970 IC50 = 65 nM T31309 CCN32L 70687971 IC50 = 700 nM T31309 CJR4L6 70687978 IC50 = 120 nM T31309 C2A8PT 70689990 IC50 = 61 nM T31309 CC4E1T 70689991 IC50 = 1790 nM T31309 CK26AI 70689992 IC50 = 100 nM T31309 CJK6O0 70689993 IC50 = 6 nM T31309 C0AL5K 70690001 IC50 = 430 nM T31309 C7WQ1I 70690002 IC50 = 160 nM T31309 COI13D 70690003 IC50 = 910 nM T31309 C7ERL2 70690004 IC50 = 32 nM T31309 CHW46I 70690005 IC50 = 710 nM T31309 CF43BG 70692160 IC50 = 110 nM T31309 CACR07 70692161 IC50 = 400 nM T31309 C2WX0B 70692162 IC50 = 15 nM T31309 CFO0R7 70692163 IC50 = 78 nM T31309 CG10VQ 70692164 IC50 = 22 nM T31309 CRAI92 70694200 IC50 = 660 nM T31309 C4OFB8 70694201 IC50 = 130 nM T31309 CG6Z3T 70694202 IC50 = 7 nM T31309 C16TJP 70694203 IC50 = 20 nM T31309 CWBC96 70694204 IC50 = 14 nM T31309 CY4B1M 70694205 IC50 = 24 nM T31309 C38ZQO 70694215 IC50 = 110 nM T31309 CAN0R1 70694216 IC50 = 32 nM T31309 CIJX30 70694217 IC50 = 140 nM T31309 CMO3U8 70694218 IC50 = 47 nM T31309 C7VY3B 70696312 IC50 = 11 nM T31309 CR56GE 70696317 IC50 = 150 nM T31309 CI4DG1 70696318 IC50 = 280 nM T31309 CY39FW 70696319 IC50 = 120 nM T31309 CH3TN5 71297204 IC50 = 5000 nM T31309 CW14HE 71449846 Ki = 3.8 nM T31309 CP45GS 71449847 Ki = 31.3 nM T31309 C1ZQ3W 71449856 Ki = 197 nM T31309 C82KST 71451661 Ki = 2.1 nM T31309 C3I5UD 71451662 Ki = 1.7 nM T31309 CQ8F0C 71451668 Ki = 178 nM T31309 C03FOT 71451669 Ki = 420 nM T31309 C8C7FS 71451698 EC50 = 3500 nM T31309 CD1N9X 71452025 Ki = 44 nM T31309 CU59ZI 71452026 Ki = 132 nM T31309 C91BPJ 71453493 Ki = 2.4 nM T31309 C4EVX6 71453494 Ki = 7.5 nM T31309 CG3C9O 71453495 Ki = 522 nM T31309 CE8B3K 71453496 Ki = 218 nM T31309 C1Q0AE 71453503 Ki = 160 nM T31309 CD52FS 71453504 Ki = 494 nM T31309 CW4J8S 71453826 Ki = 71 nM T31309 CKW71O 71455205 Ki = 39.2 nM T31309 C4QJ9E 71455206 Ki = 1.8 nM T31309 C01ZVI 71455214 Ki = 253 nM T31309 C3AS1J 71455215 Ki = 65.8 nM T31309 CPJ48S 71455216 Ki = 151 nM T31309 CJA8N4 71455243 EC50 = 9200 nM T31309 COH24E 71455246 EC50 = 6600 nM T31309 CVC5F8 71455247 EC50 = 1400 nM T31309 C2NGM3 71456995 Ki = 1.2 nM T31309 CD31ZQ 71456996 Ki = 1.7 nM T31309 C6GRP3 71456997 Ki = 569 nM T31309 CY61DU 71457007 Ki = 171 nM T31309 CGRB05 71458860 Ki = 0.8 nM T31309 CY65LH 71458861 Ki = 14.1 nM T31309 CW76ZR 71458867 Ki = 207 nM T31309 C3TL5D 71459209 Ki = 87 nM T31309 CS69ET 71459210 Ki = 24 nM T31309 CZ94MJ 71460670 Ki = 20 nM T31309 CSJ36M 71460671 Ki = 658 nM T31309 CFDQ79 71460672 Ki = 214 nM T31309 CUG8N7 71462421 EC50 = 2700 nM T31309 CVX2N9 71527715 IC50 > 4000 nM T31309 C85RZC 71527839 IC50 = 68 nM T31309 C2DZV1 71527840 IC50 = 25 nM T31309 C61XFU 71527971 IC50 < 5 nM T31309 C2Z8GU 71527972 IC50 = 25 nM T31309 CVF0O2 71545164 Ki = 9700 nM T31309 C4E1FO 71545167 Ki = 4300 nM T31309 CAW6K1 71545330 Ki = 9100 nM T31309 CHPJ72 71545486 Ki = 5300 nM T31309 CS92IM 71545651 Ki = 1400 nM T31309 CC7I6A 71545824 Ki = 960 nM T31309 CGL67T 71545826 Ki = 7400 nM T31309 CBW68J 71545828 Ki > 15000 nM T31309 CS14HM 71545993 Ki = 800 nM T31309 C0HP4B 71545994 Ki = 960 nM T31309 CP3Y2O 71548702 Ki = 6110 nM T31309 CS02CG 71549001 Ki = 7850 nM T31309 C37AJW 71549412 Ki = 23840 nM T31309 C3LIN4 71565985 Ki = 6 nM T31309 CTH79R 71605747 IC50 = 7.5 nM T31309 CZ4BU0 71605927 IC50 = 260 nM T31309 CG8Z1K 71605928 IC50 = 271 nM T31309 CAZ2N3 71605929 IC50 = 17 nM T31309 CY7L5E 71606084 IC50 = 1.1 nM T31309 C6UVA9 71606085 IC50 = 1.5 nM T31309 CR3ZA7 71606086 IC50 = 46 nM T31309 C7XK8P 71606257 IC50 = 210 nM T31309 C9G6DT 71606258 IC50 = 5.4 nM T31309 C6K8BA 71606424 IC50 = 10 nM T31309 CK1C8L 71606584 IC50 = 23 nM T31309 CJX1Y4 71624427 IC50 = 19 nM T31309 CW3QY0 71654876 Ki = 1.3 nM T31309 CU6X2Z 71656178 Ki = 59 nM T31309 CCI0N7 71656179 Ki < 0.1 nM T31309 CYFW14 71716172 IC50 = 142 nM T31309 CN2F9Z 71716725 IC50 = 2200 nM T31309 C9WS6R 71716944 IC50 = 33 nM T31309 CN86BR 71717322 IC50 = 2100 nM T31309 C5Z2XG 71717402 IC50 = 8500 nM T31309 CW4DP2 71719220 IC50 = 32 nM T31309 CNH94Q 71719979 IC50 = 35 nM T31309 CVQ6G2 71720436 IC50 = 46 nM T31309 CY08LQ 73174373 Ki = 9000 nM T31309 CO6E8W 73213478 Ki = 4600 nM T31309 CDO87T 73213545 Ki = 550 nM T31309 C9G8FB 73213546 Ki = 830 nM T31309 C90NSV 73214548 Ki = 930 nM T31309 C7O1BG 73347486 IC50 = 5000 nM T31309 CZ7SP9 73347969 Ki = 1925 nM T31309 C4L1GZ 73347970 Ki = 1323 nM T31309 CVC6Z1 73349009 IC50 > 10000 nM T31309 C6KWN5 73349012 IC50 > 10000 nM T31309 CGRZ30 73349519 Ki = 8040 nM T31309 C3TV6U 73349611 IC50 = 3.3 nM T31309 CY7KD2 73351068 Ki = 959 nM T31309 C7Q3SW 73351069 Ki = 179 nM T31309 C6ZGJ8 73353547 IC50 > 10000 nM T31309 CCH83V 73356255 IC50 = 11 nM T31309 C56WFQ 73357106 Ki = 1113 nM T31309 CR2TL5 85468775 Ki = 56 nM T31309 C3C7QO 86765310 Ki = 7560 nM T31309 CMC8E7 90478312 Ki = 1600 nM T31309 CF06DQ 90478313 Ki = 2000 nM T31309 CZ7T8W 90478318 Ki = 1600 nM T31309 CEK6S7 90478319 Ki = 1900 nM T31309 CMP47T 90478320 Ki = 2000 nM T31309 C12JEQ 91754241 Ki = 7300 nM T31309 C5T9WD 94962278 Ki = 7000 nM T31309 C20WCK 102360805 Ki = 1800 nM T31309 CHL0X1 118394626 Ki = 690 nM T31309 CO40GK 118394721 Ki = 770 nM T31309 CE28ZO 118394843 Ki = 990 nM T31309 C3BQH4 118394951 Ki = 630 nM T31309 CQT5W4 118406840 Ki = 550 nM T31309 CY1L9S 118406932 Ki = 250 nM T31309 CBTM73 118406950 Ki = 520 nM T31309 CA7DW1 118406955 Ki = 580 nM T31309 CEOY82 118406960 Ki = 950 nM T31309 CW4K9Y 118406985 Ki = 490 nM T31309 CPN23M 118406995 Ki = 140 nM T31309 CR4K9M 118705735 IC50 < 10 nM T31309 C2Q7JN 118705736 IC50 = 26 nM T31309 C23NUF 118705737 IC50 = 40 nM T31309 C27WRY 118705738 IC50 < 10 nM T31309 CT09UA 118705739 IC50 < 10 nM T31309 CN6T8R 118705740 IC50 < 10 nM T31309 CA6X5L 118705741 IC50 = 4 nM T31309 C9I0TA 118705742 IC50 < 10 nM T31309 C5G7LA 118707175 IC50 = 19 nM T31309 CD3K7L 118707176 IC50 > 1000 nM T31309 C2R8UD 118707281 IC50 = 270 nM T31309 C37IQC 118707282 IC50 = 18 nM T31309 CKN64C 118707283 IC50 = 119 nM T31309 CR1Y9J 118707284 IC50 > 468 nM T31309 CP70CG 118707285 IC50 > 1100 nM T31309 CJ9D4H 118707286 IC50 = 54 nM T31309 CI7D3R 118707287 IC50 = 250 nM T31309 CU0ZT2 118707288 IC50 = 65 nM T31309 CF4LD2 118707289 IC50 = 61 nM T31309 C6LV2K 118707290 IC50 = 19 nM T31309 COU9T1 118707291 IC50 = 545 nM T31309 CTX75Y 118707292 IC50 = 87 nM T31309 C1LD3P 118707293 IC50 < 10 nM T31309 CI5OV2 118707294 IC50 < 10 nM T31309 CO1GM8 118707295 IC50 = 17 nM T31309 C6FM7I 118707296 IC50 = 59 nM T31309 CFG28Y 118707297 IC50 = 21 nM T31309 CSE54F 118728679 Ki = 540 nM T31309 C1QW4O 118728680 Ki = 390 nM T31309 C8XBN6 118728695 Ki = 490 nM T31309 CM2B9A 118734788 Ki > 100000 nM T31309 CF73NP 118734789 Ki > 100000 nM T31309 C5W2EA 118734957 Ki > 660 nM T31309 C40BQS 118737143 Ki = 3100 nM T31309 C9BJR5 118737144 Ki = 5700 nM T31309 CNW6B0 118737146 Ki = 9900 nM T31309 CLV10W 118737147 Ki = 16000 nM T31309 CW29QH 118737148 Ki = 11700 nM T31309 CRE89M 118737149 Ki = 3700 nM T31309 C51KLE 118737150 Ki = 1100 nM T31309 C0EA6G 118737151 Ki = 4400 nM T31309 CPS8Z2 118737152 Ki = 6300 nM T31309 CQ8M7Y 118737153 Ki = 2300 nM T31309 CN7ZE6 118737156 Ki = 3700 nM T31309 CP9MA5 118737157 Ki = 770 nM T31309 C2FOD3 118737158 Ki = 1300 nM T31309 COMW16 122193136 Ki > 10000 nM T31309 CUX2N7 122193137 Ki = 900 nM T31309 CNQZ48 122193138 Ki = 7600 nM T31309 CRG62H 122193139 Ki > 10000 nM T31309 CT5N8K 122193140 Ki = 9600 nM T31309 C7RQ6J 122193141 Ki > 10000 nM T31309 C59PBG 122193142 Ki > 10000 nM T31309 C8F0MT 122193143 Ki > 10000 nM T31309 C3VSU6 122193144 Ki > 10000 nM T31309 CDJE95 122193145 Ki = 610 nM T31309 C5S6PU 122193146 Ki = 4300 nM T31309 CQ0D6T 122193147 Ki > 10000 nM T31309 CVD69Z 122193148 Ki > 10000 nM T31309 C4IUG1 122193509 Ki > 50000 nM T31309 CB9HL7 122193510 Ki > 50000 nM T31309 CIYW19 122193511 Ki > 50000 nM T31309 CV6N2D 122194465 Ki > 50000 nM T31309 CPZ09R 122194466 Ki > 50000 nM T31309 CP1WZ9 122194467 Ki > 50000 nM T31309 CQS93O 122194468 Ki > 50000 nM T31309 C0UP6Z 122194469 Ki > 50000 nM T31309 CORV91 122194470 Ki > 50000 nM T31309 C21YJS 122194471 Ki > 50000 nM T31309 CL3T2K 122194472 Ki > 50000 nM T31309 CP8EO0 122194473 Ki = 19000 nM T31309 CO5Q2K 122194474 Ki > 50000 nM T31309 CA0KR9 122194475 Ki = 3700 nM T31309 C4ODZ9 122194476 Ki = 15000 nM T31309 CJX20V 122194477 Ki > 50000 nM T31309 CXTI31 122194478 Ki = 13000 nM T31309 CM7Y4S 122194479 Ki = 4400 nM T31309 CA45FG 122194480 Ki = 13000 nM T31309 CVX9P8 122194481 Ki > 50000 nM T31309 CB8K3Q 122194482 Ki > 50000 nM T31309 CAV4M0 122194483 Ki > 50000 nM T31309 C6U2VM 122194484 Ki > 50000 nM T31309 C1Z8EY 122194485 Ki > 50000 nM T31309 CM30EU 122194486 Ki > 50000 nM T31309 C6NFG3 122194627 Ki > 10000 nM T31309 C2WX7U 122194628 Ki > 10000 nM T31309 CQ9YK2 122194629 Ki > 10000 nM T31309 C94LSC 122194630 Ki = 9000 nM T31309 C8R5NJ 122194631 Ki > 10000 nM T31309 C9SRV7 122194632 Ki = 3100 nM T31309 C46GLN 122194633 Ki > 10000 nM T31309 CUI60T 122194634 Ki = 2000 nM T31309 CNK8M7 122194635 Ki = 1600 nM T31309 C93PVM 122194636 Ki = 10000 nM T31309 CG29IZ 122194637 Ki > 10000 nM T31309 C0ZU1Y 122194638 Ki > 10000 nM T31309 CP0H3C 122194639 Ki > 10000 nM T31309 CCUF07 122194640 Ki = 3100 nM T31309 C2RA7Q 122194641 Ki > 10000 nM T31309 C5DYJ9 122194642 Ki > 10000 nM T31309 CUZV21 122194643 Ki > 10000 nM T31309 CS2GE7 122194644 Ki > 10000 nM T31309 CR19KU 122622656 Ki > 25000 nM T31309 CE4MG7 122622800 Ki > 25000 nM T31309 CBFO10 122622827 Ki = 11700 nM T31309 CY9OL2 122623097 Ki = 5600 nM T31309 C1R4UJ 122633925 Ki = 16100 nM T31309 CIBD06 127044491 Ki = 1300 nM T31309 C7KGI0 127044661 Ki = 4600 nM T31309 C63PWT 127045713 Ki = 855 nM T31309 CU75LD 127045714 Ki = 406 nM T31309 CV4K2N 127045715 Ki = 28 nM T31309 C9TS4I 127045716 Ki = 1040 nM T31309 CUT8S3 127045927 Ki = 140 nM T31309 CVEJ14 127046716 Ki = 1400 nM T31309 C4F2JM 127046867 Ki > 10000 nM T31309 C8R2OD 127046868 Ki > 10000 nM T31309 CW7KI2 127046869 Ki = 5160 nM T31309 CZ8C3V 127047003 Ki > 10000 nM T31309 C4D6XB 127047004 Ki > 10000 nM T31309 CL68JY 127047005 Ki = 694 nM T31309 CX6WE4 127047006 Ki = 932 nM T31309 C9FMI6 127047007 Ki = 5250 nM T31309 C9TCV7 127047008 Ki = 385 nM T31309 CAY7Q9 127050688 Ki = 530 nM T31309 CX3B8N 132961368 Ki > 10000 nM T31309 C81IYU 134131766 Ki = 1700 nM T31309 C2CH6A 134133054 Ki = 510 nM T31309 CBZ96D 134133726 Ki = 4900 nM T31309 CFR14T 134134268 Ki = 680 nM T31309 CJ7RT9 134135886 Ki = 2600 nM T31309 C0MAL5 134137174 Ki = 1300 nM T31309 C1D4WS 134137526 Ki = 4200 nM T31309 C91HZY 134139104 Ki = 600 nM T31309 C9YDM6 134139400 Ki = 750 nM T31309 C9ME1S 134140038 Ki = 3100 nM T31309 CM0X8W 134141608 Ki = 1900 nM T31309 CSFE39 134144182 Ki = 1500 nM T31309 C0SLU6 134148123 Ki = 3400 nM T31309 C1UHN8 134151998 Ki = 930 nM T31309 C2VC8J 134152063 Ki = 4000 nM T31309 C7ZH8I 134152922 Ki = 1700 nM T31309 CW4EP2 134153984 Ki = 4400 nM T31309 CDUI74 134154308 Ki = 670 nM T31309 C9ATX6 134154502 Ki = 1700 nM T31309 CQ24RE 134154949 Ki = 1100 nM T31309 CZ9Q5K 134155175 Ki = 1300 nM T31309 C61URW 134155768 Ki = 2000 nM T31309 CFG1Z7 134157505 Ki = 720 nM T31309 C2INR6 134828256 Ki = 730 nM T31309 CSDR07 135157296 IC50 = 495 nM T31309 C4FT3N 135403794 Ki = 286 nM T31309 CWJ5L4 135484514 IC50 = 4000 nM T31309 CAV6J3 135741996 IC50 = 170 nM T31309 C9MFV2 136002682 Ki = 140 nM T31309 C6FY0E 136002684 Ki = 150 nM T31309 CU0YE2 136032534 Ki = 1530 nM T31309 CASH13 136032535 Ki = 4470 nM T31309 C9RD0X 136032611 Ki = 230 nM T31309 CH1J4T 136126562 Ki = 224 nM T31309 CC09EN 136183442 Ki = 2080 nM T31309 CYJD84 136183443 Ki = 1450 nM T31309 CF8HV7 136183446 Ki = 31 nM T31309 C9TM5X 136190478 IC50 = 198 nM T31309 C1P6OX 136190479 IC50 = 49 nM T31309 C7QX1I 136190480 IC50 = 42 nM T31309 CM3W4P 136196528 Ki = 171 nM T31309 C6DTX1 136217518 IC50 = 96 nM T31309 CNY2V7 136217519 IC50 > 10000 nM T31309 CL1H4O 136217520 IC50 > 10000 nM T31309 CY31SM 136217522 IC50 = 1300 nM T31309 CQ76AY 136217524 IC50 = 190 nM T31309 C1BOF5 136217525 IC50 = 80 nM T31309 CAB04U 136217526 IC50 = 20 nM T31309 CO86YC 136217527 IC50 = 356 nM T31309 C2GM7B 136217528 IC50 = 206 nM T31309 C6P5FM 136217530 IC50 = 322 nM T31309 CO40EL 136217531 IC50 = 184 nM T31309 C4SW3Y 136244512 Ki = 9282 nM T31309 CQ5OS3 136249502 IC50 = 1430 nM T31309 CCG19P 136252244 IC50 = 57 nM T31309 C6J9MZ 136272994 IC50 = 21120 nM T31309 CE76MQ 136272995 IC50 = 29050 nM T31309 C7IRN8 136934823 Ki = 12000 nM T31309 CG25KR 136934824 Ki > 100000 nM T31309 C6OG0P 136934825 Ki > 100000 nM T31309 CN07GX 136934826 Ki > 100000 nM T31309 C8Z4PU 136934827 Ki > 100000 nM T31309 C1W4YP 136934828 Ki = 1900 nM T31309 CS6Z1D 136934829 Ki = 4200 nM T31309 CE9O5J 136934830 Ki = 33900 nM T31309 C1O2ZV 137078346 Ki = 1230.27 nM T31309 C73CEN 137243602 Ki = 207 nM T31309 CCDU12 137283305 Ki = 5 nM T31309 C3GOU1 137283377 Ki = 131 nM T31309 CPX64S 137289939 Ki = 182 nM T31309 C1TG3H 137290260 Ki = 235 nM T31309 CX07FI 137300716 Ki = 348 nM T31309 C9M8EW 137300717 Ki = 90 nM T31309 C28KCE 137631924 Ki = 730 nM T31309 CLP4D9 137631972 Ki = 560 nM T31309 C6EQI5 137632635 IC50 = 3830 nM T31309 CGY4X3 137632987 Ki > 10000 nM T31309 CFU98I 137634219 Ki = 920 nM T31309 C4V1YW 137634285 Ki > 10000 nM T31309 C0MNE4 137634568 Ki = 230 nM T31309 C2Z7RY 137634866 Ki > 10000 nM T31309 CKF09I 137634986 Ki = 310 nM T31309 C4IAS8 137634991 Ki > 10000 nM T31309 C53MLR 137635131 Ki > 10000 nM T31309 CU9H2I 137635438 Ki > 10000 nM T31309 C26NRZ 137635896 Ki = 580 nM T31309 CG2NQ8 137635940 Ki = 2600 nM T31309 CZ13DC 137636022 Ki = 830 nM T31309 CQ2A1K 137636996 Ki = 910 nM T31309 CI37UO 137637760 Ki > 10000 nM T31309 C9NA8L 137637871 Ki = 1300 nM T31309 CD59HQ 137638062 Ki = 270 nM T31309 CO80ZG 137638297 Ki > 10000 nM T31309 CYUH68 137639245 Ki = 470 nM T31309 C2OZJ8 137639353 Ki > 10000 nM T31309 CY25PO 137639884 Ki > 10000 nM T31309 CM4ON9 137639914 Ki > 10000 nM T31309 C42AEK 137640561 Ki = 910 nM T31309 C49LFT 137640943 Ki = 1240 nM T31309 C8F9NV 137640965 Ki > 10000 nM T31309 CTX58M 137641044 Ki = 260 nM T31309 C8HX4K 137641531 Ki > 10000 nM T31309 CGA35P 137641809 Ki = 530 nM T31309 CUPA80 137641828 Ki = 1050 nM T31309 C4MY3E 137642499 Ki > 10000 nM T31309 C37BPQ 137643293 Ki = 1410 nM T31309 CK04IH 137643542 Ki > 10000 nM T31309 CBY3S6 137644084 Ki = 740 nM T31309 C17ICS 137644285 Ki = 720 nM T31309 CGH72F 137644409 Ki = 910 nM T31309 C49CIF 137644425 Ki > 10000 nM T31309 C9XL2N 137645105 Ki > 10000 nM T31309 CR1TH2 137645619 Ki > 10000 nM T31309 C6ZIY9 137647191 Ki = 140 nM T31309 CRB6Q3 137647824 Ki = 350 nM T31309 C0J7UQ 137648092 Ki = 170 nM T31309 CL0T4U 137648463 Ki = 720 nM T31309 CRSD67 137648621 Ki > 10000 nM T31309 CQ26FC 137649261 Ki > 10000 nM T31309 C0BA4W 137650232 Ki > 10000 nM T31309 C1PLE5 137650857 IC50 = 660 nM T31309 C5TKW1 137652728 Ki > 10000 nM T31309 CH6N0I 137653797 Ki > 10000 nM T31309 CX9A0P 137654155 Ki = 440 nM T31309 C9ODE7 137654292 Ki = 810 nM T31309 CL3VX0 137655671 Ki > 10000 nM T31309 CEA7W8 137655782 Ki > 10000 nM T31309 CV9JQ2 137655840 Ki > 10000 nM T31309 CX04FN 137656103 Ki = 1190 nM T31309 C4HI7J 137656688 Ki = 5600 nM T31309 C7CWL0 137657163 Ki > 10000 nM T31309 CX87VH 137657686 Ki = 760 nM T31309 CNXE01 137658812 Ki > 10000 nM T31309 CHYZ26 137658993 Ki = 410 nM T31309 CF2SM6 137659638 IC50 = 1240 nM T31309 CEI01A 137659916 Ki > 10000 nM T31309 CDQ5I7 137660190 Ki = 750 nM T31309 C0R5IX 137660420 Ki = 150 nM T31309 CI2YP8 137660558 Ki > 10000 nM T31309 C2KN4Y 137660698 Ki > 10000 nM T31309 CAW14D 137660723 Ki > 10000 nM T31309 CP5U6T 137661597 Ki = 470 nM T31309 CNR17U 137661896 Ki = 850 nM T31309 CXH2A6 137662002 Ki > 10000 nM T31309 CWJ80Q 137662092 Ki > 10000 nM T31309 C0PQM2 138393393 IC50 = 500 nM T31309 CU91YL 138393395 IC50 = 1300 nM T31309 C5I8TQ 138756809 Ki = 28000 nM T31309 CKC68Y 139035047 IC50 = 4940 nM T31309 CP7X6U 139035048 IC50 = 540 nM T31309 C1G3HA 141721113 Ki = 630 nM T31309 CJ24FY 141721128 Ki = 500 nM T31309 CS5M3A 141721326 Ki = 380 nM T31309 CPC2E8 141733220 Ki = 560 nM T31309 C50TGO 141733221 Ki = 850 nM T31309 CY35ER 141733223 Ki = 700 nM T31309 CA40OL 141733224 Ki = 450 nM T31309 CN2TA8 141733227 Ki = 1100 nM T31309 CKJ7S9 141733229 Ki = 1500 nM T31309 CR7X5E 141733230 Ki = 570 nM T31309 CV8LZ4 141733231 Ki = 620 nM T31309 CF54KE 141733232 Ki = 580 nM T31309 C0X5YL 141733235 Ki = 5200 nM T31309 C6WJ2B 141733248 Ki = 580 nM T31309 CTR98A 141733249 Ki = 450 nM T31309 CI8J3D 145712375 IC50 = 3180 nM T31309 CMBT97 145712377 IC50 = 4780 nM T31309 C89JBL 145949373 Ki > 23000 nM T31309 C1RH9D 145950508 Ki = 1820 nM T31309 C3Y2MT 145950725 Ki > 23000 nM T31309 C01PGN 145951197 Ki = 90 nM T31309 CG1U0T 145951885 Ki = 620 nM T31309 C4JY1B 145951938 Ki > 23000 nM T31309 C13BLU 145952150 Ki > 23000 nM T31309 CJ9RW7 145952398 Ki = 1450 nM T31309 CMP86N 145952997 Ki > 23000 nM T31309 CR86NC 145953250 Ki = 830 nM T31309 CDRT57 145953525 Ki > 23000 nM T31309 C15HUW 145953591 Ki = 2220 nM T31309 C8VIT4 145954556 Ki > 23000 nM T31309 CKM98O 145954557 Ki > 23000 nM T31309 C6C9UX 145955049 Ki > 23000 nM T31309 C3YPX4 145955393 Ki = 320 nM T31309 CT32ER 145955454 Ki > 23000 nM T31309 C0DFZ5 145956250 Ki = 1080 nM T31309 CXA7J4 145956350 Ki > 23000 nM T31309 CPWL30 145956560 Ki > 23000 nM T31309 CQ56PE 145956913 Ki > 23000 nM T31309 C5VPR7 145957258 Ki > 23000 nM T31309 CTLC26 145958175 Ki = 370 nM T31309 C6ZH2C 145958475 Ki = 450 nM T31309 CDJL71 145958776 Ki > 23000 nM T31309 CH23LV 145958880 Ki > 23000 nM T31309 C40QTV 145959015 Ki > 23000 nM T31309 CC82IQ 145959586 Ki = 2580 nM T31309 C7NH1G 145960303 Ki = 3600 nM T31309 CBEH81 145964348 IC50 = 17.3 nM T31309 CL7K3I 145965147 IC50 = 68.2 nM T31309 CB7G6P 145965660 IC50 = 46 nM T31309 CG7P1Z 145966192 IC50 = 57.9 nM T31309 C2RJ4H 145966654 IC50 = 65.1 nM T31309 C5SN3Q 145966763 IC50 = 168 nM T31309 CNSQ67 145967322 IC50 = 40.7 nM T31309 C3XRD8 145967779 IC50 = 108 nM T31309 C5FL7B 145968700 IC50 = 67.4 nM T31309 CB5O9E 145971233 Ki = 700 nM T31309 CH51QR 145972482 Ki = 1540 nM T31309 CGAZ83 145972946 Ki = 1420 nM T31309 C7R5ED 145973286 IC50 = 12.6 nM T31309 C37LPJ 145973505 IC50 = 38.1 nM T31309 CYQR17 145973714 IC50 = 193 nM T31309 CU65EX 145974322 Ki = 2920 nM T31309 CM6U1R 145976325 IC50 > 1000 nM T31309 CD8Q9R 145976379 IC50 = 46.6 nM T31309 C52PKW 145977421 IC50 = 14.5 nM T31309 C2QPU1 145977736 IC50 = 34.8 nM T31309 C9LBE6 145978364 IC50 = 20.7 nM T31309 CL76CK 145978956 IC50 = 50.1 nM T31309 CKF3S0 145979166 IC50 = 2.8 nM T31309 CGIZ51 145979582 IC50 = 9.7 nM T31309 CZUD98 145979683 IC50 = 86.5 nM T31309 CL0H3M 145979783 IC50 = 3.5 nM T31309 C0NJC3 145982309 IC50 = 34.7 nM T31309 CG4QD0 145983256 Ki = 610 nM T31309 C6UVF9 145984310 Ki = 880 nM T31309 CT2KN0 145984576 Ki = 800 nM T31309 CURF95 145984861 Ki = 390 nM T31309 CP39XU 145985660 IC50 = 11.9 nM T31309 CI6K3W 145986491 IC50 = 6.2 nM T31309 CU9I4K 145989784 IC50 = 31.9 nM T31309 C7WT5C 145989980 IC50 = 16.7 nM T31309 CSZ4M5 145990737 IC50 = 5 nM T31309 CTVC87 145991099 IC50 = 1.8 nM T31309 CQ8M0P 145991800 IC50 = 13 nM T31309 C4BM9U 145991913 IC50 = 1.9 nM T31309 C2OG0L 145993372 IC50 = 67.1 nM T31309 C9KI8G 145993554 IC50 = 28.7 nM T31309 C0NWC7 145993811 IC50 = 2.2 nM T31309 CW4O5A 145993860 IC50 = 1.2 nM T31309 CCVP03 145994390 Ki > 25000 nM T31309 CZ0KI3 155511427 Ki > 5000 nM T31309 CL9HJ7 155511905 IC50 = 11650 nM T31309 C59APO 155513041 Ki = 4900 nM T31309 CK25AN 155513849 Ki = 440 nM T31309 CBG8V7 155513976 Ki = 470 nM T31309 C9Z8FQ 155514893 Ki = 359000 nM T31309 C0RY3A 155514968 Ki = 560 nM T31309 CTE3V7 155515598 Ki = 51000 nM T31309 CJ7A1D 155516576 Ki = 49000 nM T31309 C3X0SP 155518228 Ki = 1300 nM T31309 CB37YD 155518816 IC50 > 99000 nM T31309 CKPO27 155518834 Ki > 5000 nM T31309 C91LSI 155520022 Ki = 21000 nM T31309 CUJY40 155521076 Ki = 24000 nM T31309 CE6QM8 155522510 Ki = 36000 nM T31309 CQ6A8T 155524065 IC50 = 10480 nM T31309 C3HYI9 155524558 Ki = 470000 nM T31309 C6W9LH 155524710 Ki = 8100 nM T31309 C9J0YL 155524932 IC50 = 15210 nM T31309 CNH49E 155525790 Ki = 510 nM T31309 C01CQS 155526457 Ki = 418000 nM T31309 CXY0L3 155527670 Ki = 13000 nM T31309 CHA14B 155527900 Ki = 437000 nM T31309 CT6M0W 155530529 Ki = 630 nM T31309 CF2KP7 155530563 Ki = 5400 nM T31309 CJS3M8 155531324 Ki > 5000 nM T31309 C95XMJ 155532216 Ki = 6100 nM T31309 CQ68DY 155533068 Ki > 5000 nM T31309 CK6W2Y 155534018 IC50 = 240 nM T31309 C7L8AM 155534540 IC50 = 2310 nM T31309 C4ZNJ7 155534814 Ki = 269000 nM T31309 C2ME5X 155534955 Ki > 5000 nM T31309 CV3L8Q 155536071 Ki = 4100 nM T31309 CNAR96 155536134 IC50 = 27600 nM T31309 CE98TA 155536902 Ki > 5000 nM T31309 CW5G2H 155537202 Ki = 560 nM T31309 CK7UQ4 155537237 IC50 = 1300 nM T31309 C0VBW2 155538516 IC50 = 13470 nM T31309 CEAJ80 155539156 Ki = 24000 nM T31309 C6NI9J 155539696 Ki = 450 nM T31309 C5HAC4 155539927 Ki = 430 nM T31309 CW1EL8 155539938 Ki = 29000 nM T31309 C8K0QO 155541624 Ki = 520 nM T31309 C2ICU5 155541804 IC50 = 20 nM T31309 CC3A4H 155541877 Ki = 310 nM T31309 C81PLG 155542475 Ki = 5000 nM T31309 C8CEJ5 155542773 Ki = 1300 nM T31309 CUS28M 155542793 Ki = 1200 nM T31309 CU3A9B 155543367 Ki = 0.36 nM T31309 C7IK3P 155544559 Ki = 530 nM T31309 CS0X8D 155545070 Ki > 5000 nM T31309 CI7L0N 155545489 Ki = 480 nM T31309 C6TQ4X 155545656 IC50 = 2000 nM T31309 C0A1YL 155546744 Ki = 59 nM T31309 C8PG9F 155546898 Ki > 5000 nM T31309 CL4HF7 155547093 Ki = 1200 nM T31309 C4SM7J 155547389 IC50 = 1940 nM T31309 C4LTY2 155548831 Ki = 590 nM T31309 COSN81 155549762 Ki = 670 nM T31309 CH72LS 155553237 Ki = 440 nM T31309 CE2KQ4 155555867 IC50 = 4520 nM T31309 CNPA24 155558338 IC50 = 7660 nM T31309 CUX0F2 155558443 IC50 = 55900 nM T31309 CHBE37 155560310 IC50 = 10020 nM T31309 C6JC3K 155563087 Ki = 74000 nM T31309 CYIB91 155563107 Ki = 98000 nM T31309 CG59ZN 155564461 IC50 = 9710 nM T31309 CAG01V 155565290 IC50 = 230 nM T31309 CA68BM 155565390 IC50 = 2240 nM T31309 C5Y0QF 155565915 IC50 = 9700 nM T31309 C3W7RP 155569171 IC50 = 250 nM T31309 C8CL3Z 155569283 IC50 = 6300 nM T31309 CN10OD 59053562 IC50 = 350 nM T31309 C04MNK 71527841 IC50 = 17 nM T31309 D00LHS 11455910 IC50 = 200 nM T31309 D04RTY 16090304 IC50 = 5000 nM T31309 D05RDP 992586 Ki = 2900 nM T31309 D06AQG 135468219 IC50 = 1600 nM T31309 D0D6BH 379493 IC50 = 4700 nM T31309 D0T3VP 2782689 IC50 = 300000 nM T31309 D0V7PX 454878 Ki = 640 nM T31309 D0X0CS 16090303 IC50 = 7000 nM T69208 D06KTJ 53252276 IC50 = 226 nM T69208 D0E3TC 44259 IC50 < 0.1 nM T69208 D0T3ME 156422 IC50 > 30000 nM T69208 CACS26 11561968 Ki > 2000 nM T69208 CU0E8O 11690457 Ki > 2000 nM T69208 C3VRO9 44557921 IC50 > 10000 nM T69208 CLS29B 46872626 IC50 > 10000 nM T69208 C8NA4L 53384644 IC50 > 30000 nM T69208 C8AB1J 54759606 Ki = 840 nM T69208 C1MR8Q 60097495 IC50 > 1000 nM T69208 CV63UL 67240318 IC50 > 10000 nM T69208 D0E7VO 59627005 IC50 = 6.1 nM T99189 D00JAU 3749 IC50 = 30000 nM T99189 D02ZTJ 5339 IC50 = 9600 nM T99189 D05DVP 5717 IC50 = 6500 nM T99189 D08GHB 446155 IC50 = 40000 nM T99189 D0S7JH 16004692 IC50 = 10000000 nM T99189 D0U4CE 104865 IC50 = 30000000 nM T99189 D0J6XC 5803 IC50 = 6900 nM T99189 D0V1WQ 24857286 IC50 = 2000 nM T99189 CU7MI6 44392310 IC50 = 200 nM T99189 CP8IA6 44392321 IC50 = 300 nM T99189 CW4K1S 44392322 IC50 = 300 nM T99189 CI4CP8 44392323 IC50 = 8600 nM T99189 CU5W6D 44392324 IC50 = 63000 nM T99189 CJ42NL 44392345 IC50 = 3400 nM T99189 C45YDE 44392346 IC50 = 220 nM T99189 CMT2Q5 44392360 IC50 = 1600 nM T99189 CK1J8G 44392368 IC50 = 300 nM T99189 CIJ5C2 44392375 IC50 = 700 nM T10491 C3DM0P 1509257 IC50 = 10000 nM T10491 CIAX42 1907637 IC50 = 5360 nM T10491 CQBT36 3170817 IC50 = 9790 nM T10491 CTC2F6 3377049 IC50 = 1290 nM T10491 C8A4YP 4907613 IC50 = 1490 nM T10491 CM9NV7 4915043 IC50 = 8020 nM T10491 CI2U6Q 4919494 IC50 = 4350 nM T10491 CFO5K6 9890095 Ki = 15.85 nM T10491 C5TWF9 10055825 IC50 > 30000 nM T10491 CF8KR4 10073347 Ki = 398.11 nM T10491 CWF87Z 10078747 IC50 = 18000 nM T10491 CL2HO4 10093732 Ki = 25.12 nM T10491 C1W4TD 10431044 Ki = 1584.89 nM T10491 CR2J6L 10485171 IC50 > 30000 nM T10491 CAKI94 16020224 IC50 = 2210 nM T10491 CMPQ63 16102648 EC50 = 74 nM T10491 C0UZN8 16102649 IC50 = 13000 nM T10491 CWQ03V 16102650 IC50 = 4600 nM T10491 C0EKY9 16102652 IC50 > 30000 nM T10491 CD51PH 16102653 IC50 > 30000 nM T10491 C73TRI 17016126 IC50 = 1870 nM T10491 CJX4L9 20861881 IC50 = 2160 nM T10491 CEQP65 20873176 IC50 = 11400 nM T10491 CEXW20 20879988 IC50 = 7000 nM T10491 CN7SO4 20940584 IC50 = 3890 nM T10491 C7W4CX 20940617 IC50 = 3200 nM T10491 C26TEQ 20940674 IC50 = 6750 nM T10491 CDM5Z4 22514197 IC50 = 2780 nM T10491 CI80AS 23602867 IC50 = 6330 nM T10491 C71DKT 23602886 IC50 = 5270 nM T10491 C7QJ1Y 40136736 IC50 = 5840 nM T10491 CB9JF5 42700768 Ki = 199.53 nM T10491 C9A6QF 46202768 IC50 < 100 nM T10491 C58LCB 46250897 IC50 = 6190 nM T10491 C82LCD 46273745 IC50 = 2640 nM T10491 CP81MI 46503468 IC50 = 2920 nM T10491 C4BP7N 53355383 EC50 = 31.62 nM T10491 CXMJ34 59004228 IC50 < 1000 nM T10491 CRC03O 59052012 Ki = 12.59 nM T10491 CV14CL 59052013 Ki = 794.33 nM T10491 CT6FB1 59052014 Ki = 1258.93 nM T10491 CF3GA4 59052140 Ki = 794.33 nM T10491 CT0G2U 59052141 Ki = 794.33 nM T10491 CAK79I 59052142 Ki = 31.62 nM T10491 CW7K6E 59052143 Ki = 100 nM T10491 CU2DH8 59052144 Ki = 50.12 nM T10491 CLZA71 59052145 Ki = 79.43 nM T10491 C08ZFS 59052281 Ki = 79.43 nM T10491 CBZ4O1 59052282 Ki = 100 nM T10491 CQ3BP8 59052283 EC50 = 1400 nM T10491 C58EOU 59052284 Ki = 5011.87 nM T10491 CUH0K2 59052285 EC50 = 1.6 nM T10491 C5RQE0 59052424 EC50 = 1 nM T10491 CH1QI4 59052425 Ki = 1258.93 nM T10491 CW6ZR8 59052426 Ki = 1258.93 nM T10491 CDNH85 59052427 Ki = 1584.89 nM T10491 C06CAJ 59052428 Ki = 3162.28 nM T10491 C6E5UG 59366166 Ki = 7.943 nM T10491 C4QI3R 70809652 Ki = 18000 nM T10491 C5HP1T 73351942 IC50 = 4740 nM T10491 C6ENV5 100951623 IC50 > 10000 nM T10491 C7W0LF 122178716 IC50 = 15000 nM T10491 CQ4Y2B 122178717 IC50 > 30000 nM T10491 C4X5HK 122178718 IC50 > 30000 nM T10491 CX0D2P 122178719 IC50 > 30000 nM T10491 CXJ01F 122178720 IC50 > 30000 nM T10491 CCZF85 122178721 IC50 = 18000 nM T10491 C1HM2J 122178722 IC50 = 2400 nM T10491 CJ5FP0 122178723 EC50 = 91 nM T10491 C5NT4D 122178724 IC50 = 3400 nM T10491 CR8AJ9 122178725 IC50 = 23000 nM T10491 CM6W9J 122178726 IC50 = 13000 nM T10491 CE1AR2 122178727 IC50 = 4600 nM T10491 CV7UY5 122178728 IC50 > 30000 nM T10491 C8EJT2 122178729 IC50 > 30000 nM T10491 CN6S8D 122178730 IC50 = 16000 nM T10491 C19BRQ 122178731 IC50 = 11000 nM T10491 CU7TK1 122178732 IC50 > 30000 nM T10491 CLD78B 134694953 EC50 = 11 nM T10491 C3SM8K 137631624 IC50 = 2600 nM T10491 C9BV5Z 137632091 Ki = 760 nM T10491 C02MSJ 137632194 IC50 = 3600 nM T10491 CA78OM 137632639 Ki = 950 nM T10491 CU1H0F 137632681 IC50 = 690 nM T10491 CJ9FM7 137632684 Ki = 1900 nM T10491 CTH4R9 137633428 Ki = 24 nM T10491 CKI7E3 137634082 IC50 = 2000 nM T10491 C1S2YN 137634372 IC50 = 2000 nM T10491 CQS70B 137634879 IC50 = 2000 nM T10491 CT8YI0 137635322 IC50 = 4100 nM T10491 C0V9CY 137636041 IC50 = 2200 nM T10491 CG84FX 137636198 IC50 = 4000 nM T10491 C8GLY9 137636313 IC50 = 2000 nM T10491 C51ALD 137636455 IC50 = 1300 nM T10491 CM9YP4 137636536 IC50 = 840 nM T10491 C6DLP5 137636611 Ki = 7943.28 nM T10491 C9ZVB0 137637180 Ki = 19.95 nM T10491 C6A4JC 137637520 IC50 = 2000 nM T10491 C4T7AF 137637674 IC50 = 4200 nM T10491 CZ2VC9 137637920 Ki = 760 nM T10491 CGX7S1 137638021 Ki = 95 nM T10491 CLCG42 137638059 IC50 = 2000 nM T10491 C49CAF 137638093 IC50 = 1000 nM T10491 CQ9PI1 137638674 IC50 = 560 nM T10491 CF8S5N 137639002 EC50 = 7 nM T10491 CTV94W 137639137 IC50 = 1800 nM T10491 CMF9Q1 137639293 IC50 = 1100 nM T10491 C5MB8S 137639423 EC50 = 46 nM T10491 CYZ70O 137639573 Ki = 23 nM T10491 C1OG4M 137640505 IC50 = 2000 nM T10491 CRVT81 137640610 Ki = 31.62 nM T10491 CB5L0M 137640842 IC50 = 4600 nM T10491 CW9Z8I 137641374 Ki = 900 nM T10491 CR0NM5 137641851 Ki = 31.62 nM T10491 CX25HG 137642442 Ki = 29 nM T10491 CWI2V7 137643302 Ki = 501.19 nM T10491 CO01IW 137643816 IC50 = 9500 nM T10491 C0UFD2 137643985 Ki = 31.62 nM T10491 C31KCL 137644260 IC50 = 850 nM T10491 CW7R9J 137644796 IC50 = 190 nM T10491 CYI0F2 137644874 IC50 = 250 nM T10491 CB78AN 137644938 IC50 = 13000 nM T10491 C78HFG 137645641 IC50 = 2000 nM T10491 C8DF4P 137645906 IC50 = 1900 nM T10491 CZC5B4 137646887 Ki = 501.19 nM T10491 C84IVY 137647312 Ki = 7.943 nM T10491 CT86OF 137647937 IC50 = 4900 nM T10491 C45BXQ 137648096 Ki = 7700 nM T10491 C4DY6Z 137648169 IC50 = 410 nM T10491 CPJV29 137648481 IC50 = 2000 nM T10491 CCT4L9 137649106 IC50 = 600 nM T10491 CKWA09 137649205 Ki = 398.11 nM T10491 C34XMR 137649383 Ki = 63.1 nM T10491 CH7MV8 137650158 IC50 = 2000 nM T10491 CRP80C 137650276 IC50 = 790 nM T10491 C84MCE 137650399 Ki > 9700 nM T10491 C3G8ZH 137650942 Ki = 9 nM T10491 CYC8B5 137651257 Ki = 199.53 nM T10491 CG17FC 137651398 Ki = 71 nM T10491 CC75QA 137651588 IC50 = 720 nM T10491 CY84HV 137651875 Ki = 39.81 nM T10491 CRH02L 137652168 IC50 = 540 nM T10491 CLI17P 137653464 Ki = 39.81 nM T10491 C2JXO5 137653472 Ki = 189 nM T10491 CMAG96 137653666 Ki = 4500 nM T10491 C9Y0QE 137654056 Ki = 730 nM T10491 CP53IG 137654154 Ki = 774 nM T10491 CV35EJ 137654804 IC50 = 2600 nM T10491 C71JBT 137655000 Ki = 30 nM T10491 CE6L3M 137655149 IC50 = 2000 nM T10491 CUC1D4 137655552 IC50 = 5800 nM T10491 C65MBR 137655630 EC50 = 110 nM T10491 C8ZOE4 137655757 Ki = 79.43 nM T10491 C5S3IL 137655887 IC50 = 2100 nM T10491 C25RWZ 137655917 IC50 = 3200 nM T10491 CRW05J 137656262 IC50 = 450 nM T10491 CNU89M 137656325 IC50 = 5000 nM T10491 C4IU6W 137656583 Ki = 5.012 nM T10491 CQJB39 137656753 Ki = 7.943 nM T10491 CB6CZ4 137656904 Ki = 12589.25 nM T10491 CN4C2T 137657155 IC50 = 350 nM T10491 CNW79C 137658328 Ki = 50.12 nM T10491 CZ70YL 137658374 IC50 = 2000 nM T10491 CPK8C1 137658844 Ki = 63 nM T10491 C9XJ5A 137659767 Ki = 96 nM T10491 C1VZ2U 137659906 IC50 = 720 nM T10491 CH9A8Q 137660298 IC50 = 520 nM T10491 CPI59B 137660618 Ki = 25 nM T10491 C1R5BU 137660760 IC50 = 1300 nM T10491 C51FPJ 137660789 IC50 = 1200 nM T10491 C9M7JB 137660814 IC50 = 2000 nM T10491 CAP85L 137660893 IC50 = 2600 nM T10491 C5Q8UM 137662063 IC50 = 1500 nM T10491 C2VRA9 137662172 IC50 = 1800 nM T10491 C6ZU0A 145949555 EC50 > 20000 nM T10491 CE3D8P 145951877 EC50 > 20000 nM T10491 CI9BO4 145952624 EC50 = 7810 nM T10491 CL42TO 145953024 EC50 = 3970 nM T10491 CR2QH0 145957924 EC50 = 5920 nM T10491 CP25CA 145958767 EC50 = 10460 nM T10491 C01GKQ 145971455 EC50 > 20000 nM T10491 CFC74M 155531067 EC50 = 690 nM T10491 C4XRZ1 155558626 EC50 = 1700 nM T10491 D04TIO 5275843 EC50 = 1995.26 nM T56367 D03VPC 2754 IC50 > 1000000 nM T56367 D05MQK 110635 IC50 > 10000 nM T56367 D06BCB 443955 Ki = 14000 nM T56367 D0C9SY 135400189 IC50 = 300 nM T56367 D0E0SW 53708 IC50 > 1000000 nM T56367 D0F8RA 2153 IC50 = 320000 nM T56367 D0F9GE 3108 IC50 = 45000 nM T56367 D0NJ3V 4680 IC50 = 9000 nM T56367 D0Y9ZE 4197 IC50 = 310000 nM T56367 D0Z7ZM 135398744 IC50 = 819 nM T56367 D0T5PO 5092 IC50 > 100000 nM T56367 D0X0PP 59351313 IC50 > 30000 nM T56367 D00SPK 23665864 IC50 = 4700 nM T56367 D00YPW 135399235 IC50 = 1100 nM T56367 D02EMR 151170 IC50 > 10000 nM T56367 D07FHZ 5087 IC50 = 250000 nM T56367 D09UMA 55918 IC50 > 1000000 nM T56367 D0BK6B 3021729 IC50 > 100000 nM T56367 D0GR2J 3034011 IC50 = 1500 nM T56367 CVQ0G5 1348 Ki = 9500 nM T56367 C03NGJ 1713 IC50 > 100000 nM T56367 CO2Y3R 3698 IC50 > 300000 nM T56367 CCJ8F0 5353 IC50 > 1000000 nM T56367 CJ02EG 41946 Ki = 10000 nM T56367 CGA17S 127779 Ki = 3700 nM T56367 C54IRL 129517 IC50 = 409000 nM T56367 CR8H1B 149028 IC50 = 1900 nM T56367 CK4VZ8 152034 IC50 = 86000 nM T56367 C0YK8A 155806 IC50 = 5200 nM T56367 COK69D 156890 IC50 = 265000 nM T56367 C78DLE 205964 IC50 = 5500 nM T56367 C4IEB6 205981 Ki = 717000 nM T56367 CO0Z8N 1002275 IC50 = 5700 nM T56367 C0JM2Q 1215407 IC50 = 1900 nM T56367 CZ2XI5 1271431 IC50 = 3700 nM T56367 C6AT3L 2930929 IC50 = 2500 nM T56367 CWO8I2 3041753 IC50 = 4400 nM T56367 CD70ZG 3119958 IC50 = 300 nM T56367 C4MSC9 3120507 IC50 = 2500 nM T56367 CC3LA4 4672917 IC50 = 890 nM T56367 C5P0LU 4672918 IC50 = 7010 nM T56367 C0C9HP 6610310 IC50 > 100000 nM T56367 CAYS61 6918354 IC50 = 2000 nM T56367 CB40PM 6918356 IC50 = 10000 nM T56367 CI7K0P 6918667 IC50 = 3260 nM T56367 CP1GO7 6918668 IC50 = 5160 nM T56367 C87WYR 6918795 IC50 = 6290 nM T56367 CRGE51 6918796 IC50 = 11600 nM T56367 CUP4M8 6918797 IC50 = 6470 nM T56367 C0LRO8 6918798 IC50 = 4760 nM T56367 C53ESK 6918799 IC50 = 10500 nM T56367 CU1E0G 6918800 IC50 = 29000 nM T56367 CRU46D 7161211 IC50 > 10000 nM T56367 CNC2F4 9798336 IC50 > 1000000 nM T56367 CFJ62Y 9799389 IC50 > 10000 nM T56367 C2FIY8 9808974 IC50 = 200 nM T56367 C1CXA5 9818702 IC50 = 40000 nM T56367 C4J2XE 9836643 IC50 > 101000 nM T56367 C8QJ4D 9859958 IC50 = 40000 nM T56367 CF18MC 9874535 IC50 = 3000 nM T56367 C0Q5VN 9880010 IC50 > 101000 nM T56367 CWD1F6 9880288 IC50 = 72400 nM T56367 C7XYK6 9881656 IC50 > 100000 nM T56367 CD6IG8 9894586 IC50 = 33000 nM T56367 CC05QE 9901606 IC50 = 85680 nM T56367 CMBO89 9912467 IC50 = 2000 nM T56367 CBA29H 9922545 IC50 = 5860 nM T56367 CKF4C2 9922691 IC50 = 33000 nM T56367 C70AMC 9924305 IC50 = 16380 nM T56367 CKI6N2 9924468 IC50 = 320 nM T56367 C6AZ5F 9924709 IC50 > 101000 nM T56367 CX1UV7 9946954 IC50 = 40340 nM T56367 C7OP5A 9947052 IC50 = 5230 nM T56367 C62RCW 9959690 IC50 = 40000 nM T56367 CJO0X4 9966737 IC50 = 9810 nM T56367 CFP1Y5 9966830 IC50 > 101000 nM T56367 C9NKY4 9967652 IC50 = 19000 nM T56367 CI6AX1 9968005 IC50 = 7830 nM T56367 C7PCS8 9968050 IC50 = 28930 nM T56367 CFB48Q 9968370 IC50 > 101000 nM T56367 CU73AJ 9968471 IC50 > 101000 nM T56367 C0AP8O 9969020 IC50 = 21580 nM T56367 C5AE2I 9973597 IC50 > 200000 nM T56367 CW3S7O 9977675 IC50 > 1000000 nM T56367 C7X0UM 9984330 IC50 = 2200 nM T56367 C9LI5W 9985050 IC50 = 1000 nM T56367 CO87TV 9994528 IC50 > 100000 nM T56367 CB9EY5 9995187 IC50 > 100000 nM T56367 C6MUC5 10024867 IC50 > 40000 nM T56367 CT6Y9J 10043209 IC50 > 1000000 nM T56367 CC6PO8 10066654 IC50 > 40000 nM T56367 C3MA2L 10067044 IC50 > 1000000 nM T56367 CI4T1D 10075879 IC50 = 1100 nM T56367 CJ16FV 10087963 IC50 > 1000000 nM T56367 CRW6E1 10088941 IC50 > 40000 nM T56367 C13QUP 10089597 IC50 = 400000 nM T56367 CARY56 10091146 IC50 > 200000 nM T56367 CG61LB 10097991 IC50 = 9 nM T56367 C12LED 10109572 IC50 > 101000 nM T56367 C2PBD6 10131447 IC50 = 2860 nM T56367 C5HC2X 10182563 IC50 = 6390 nM T56367 C3GN8K 10200432 IC50 = 1600 nM T56367 CFGO46 10221904 IC50 = 650 nM T56367 CZ1Y8D 10232923 IC50 > 100000 nM T56367 CT7RC0 10245770 IC50 = 22000 nM T56367 CP4YR0 10248176 IC50 > 1000000 nM T56367 C7MQZ1 10249183 IC50 > 1000000 nM T56367 C0PD9Y 10255798 IC50 = 2000 nM T56367 CQ61CV 10268304 IC50 = 8300 nM T56367 C1QU2B 10268305 IC50 = 3010 nM T56367 CH9C4K 10269859 IC50 = 14060 nM T56367 CR92JY 10270352 IC50 = 29700 nM T56367 C7CHR0 10270536 IC50 = 710 nM T56367 C6AQ0U 10338401 IC50 > 200000 nM T56367 C52EPV 10339653 IC50 > 1000000 nM T56367 CEIW08 10359077 IC50 > 200000 nM T56367 CB0D8J 10371031 IC50 = 300 nM T56367 C52DNX 10384462 IC50 > 40000 nM T56367 CF6A1Q 10385088 IC50 > 200000 nM T56367 CZ6X9Y 10391444 IC50 = 85 nM T56367 CUF0X6 10404302 IC50 > 1000000 nM T56367 CAW23H 10434818 IC50 > 1000000 nM T56367 CF5O8D 10446136 IC50 = 38800 nM T56367 CZ8IC4 10448177 IC50 > 1000000 nM T56367 C1RZ9E 10449000 IC50 > 1000000 nM T56367 CU2HN6 10450290 IC50 > 200000 nM T56367 C6PXC2 10471556 IC50 > 100000 nM T56367 C2DEO3 10472374 IC50 = 250000 nM T56367 C5CI3G 10479468 IC50 = 100000 nM T56367 CA24TW 10491646 IC50 > 100000 nM T56367 C68VBD 10492653 IC50 > 100000 nM T56367 C3PKX6 10492654 IC50 > 100000 nM T56367 CTUW75 10503944 IC50 = 820 nM T56367 C6GS9R 10506218 IC50 > 100000 nM T56367 CYVR93 10507187 IC50 = 800 nM T56367 C4CN0V 10508072 IC50 = 11000 nM T56367 CW7T6I 10515565 IC50 > 100000 nM T56367 CPWU60 10524067 IC50 = 30000 nM T56367 C9WSE6 10528313 IC50 > 100000 nM T56367 CZ6T2C 10536740 IC50 > 100000 nM T56367 CCG53Q 10541661 IC50 = 52000 nM T56367 CP0JT2 10550927 IC50 > 100000 nM T56367 CQW79N 10554042 IC50 > 100000 nM T56367 C4V8OI 10563356 IC50 > 100000 nM T56367 CY9P5W 10575733 IC50 > 100000 nM T56367 C7Z9YF 10579873 IC50 = 61000 nM T56367 C57HYA 10600864 IC50 = 35000 nM T56367 CS2Q1U 10602534 IC50 > 100000 nM T56367 C10QMP 10602807 IC50 = 400 nM T56367 CSPY93 10603533 IC50 = 1100 nM T56367 CJ7CU4 10603606 IC50 = 20000 nM T56367 C8P3GS 10603764 IC50 = 1200 nM T56367 C5LVM2 10613420 IC50 > 100000 nM T56367 CK3GR5 10624131 IC50 = 9000 nM T56367 CZIQ04 10625498 IC50 = 29000 nM T56367 CN4T7O 10625920 IC50 > 100000 nM T56367 C21CUM 10626417 IC50 = 89000 nM T56367 C1O4KV 10626842 IC50 = 41000 nM T56367 C25WRZ 10627119 IC50 = 4000 nM T56367 CNK65G 10646809 IC50 = 100000 nM T56367 CKNA14 10648008 IC50 = 5000 nM T56367 C3XAK7 10650055 IC50 = 88000 nM T56367 CE65JO 10650764 IC50 = 26000 nM T56367 CNP1D9 10651107 IC50 = 13000 nM T56367 CTL2D5 10651687 IC50 = 1600 nM T56367 CJ5XI4 10651803 IC50 > 100000 nM T56367 CB9Y7A 10669693 IC50 = 50000 nM T56367 CFM5N1 10673963 IC50 = 69000 nM T56367 CZ08CE 10674739 IC50 = 500 nM T56367 C9FR7P 10674875 IC50 = 13000 nM T56367 C2Y5HF 10675032 IC50 = 3000 nM T56367 CV6WT3 10692240 IC50 > 100000 nM T56367 CBW2X8 10697689 IC50 = 600 nM T56367 CI6ON5 10698519 IC50 = 2000 nM T56367 C91VBT 10699116 IC50 = 200 nM T56367 C23WGX 10706416 IC50 = 14000 nM T56367 CDMP96 10717370 IC50 = 50000 nM T56367 CCI8R7 10729204 IC50 > 100000 nM T56367 C7JN8X 10739699 IC50 = 2100 nM T56367 CINX82 10763354 IC50 > 100000 nM T56367 CLM42P 10788651 IC50 = 40000 nM T56367 C19EHR 10791038 IC50 = 77000 nM T56367 CXWY95 10792119 IC50 = 55000 nM T56367 C6C5AD 10792156 IC50 = 27000 nM T56367 C2KUF1 10792829 IC50 = 45000 nM T56367 C1K4AN 10792853 IC50 = 26000 nM T56367 C4T8PS 10816641 IC50 = 3400 nM T56367 CX1B4U 10817302 IC50 = 24000 nM T56367 CZMB59 10840332 IC50 > 100000 nM T56367 C5MTK7 10840471 IC50 > 100000 nM T56367 C2IWD7 10840815 IC50 = 3500 nM T56367 CR50XV 10841036 IC50 > 100000 nM T56367 CREQ98 11373312 IC50 = 5800 nM T56367 C45VZC 11438405 IC50 > 16000 nM T56367 C4ZYH9 11547485 IC50 > 10000 nM T56367 CM5T9U 11724564 IC50 = 20000 nM T56367 C0AKJ4 11742456 IC50 = 14000 nM T56367 CGA1F8 11794425 IC50 = 70000 nM T56367 CYX91E 11795941 IC50 = 16000 nM T56367 C30UGZ 11800567 IC50 = 74000 nM T56367 C4GK2R 11801613 IC50 = 200 nM T56367 CC6M3T 12134735 IC50 = 20 nM T56367 CE41YR 13059432 IC50 = 580000 nM T56367 CEY1B7 13066339 Ki = 4000 nM T56367 C7SPV8 13233881 IC50 > 1000000 nM T56367 C75JTV 13233882 IC50 > 1000000 nM T56367 C9NR8P 13233885 IC50 > 1000000 nM T56367 C4AK6E 13233889 IC50 = 790000 nM T56367 CZ50CU 13887375 IC50 = 330000 nM T56367 CASB70 14099426 IC50 > 1000000 nM T56367 CI3J7R 14099427 IC50 = 220000 nM T56367 CQ1LY8 14099432 IC50 = 140000 nM T56367 CUS17I 14099444 IC50 = 930000 nM T56367 CP5JU9 14099446 IC50 = 660000 nM T56367 C17HNR 14099449 IC50 > 500000 nM T56367 CR8Z4H 14403301 IC50 = 2300 nM T56367 C2ZX8H 14756622 IC50 = 820 nM T56367 CAC5H0 15606258 IC50 > 100000 nM T56367 CW6MV8 15981426 IC50 = 87 nM T56367 C3LJ4B 19003750 IC50 = 1800 nM T56367 CJ95TM 20146320 IC50 = 80000 nM T56367 C58VPG 21212519 IC50 = 2500 nM T56367 C7RK1W 21920272 IC50 = 9280 nM T56367 CH7N9S 21920275 IC50 = 3340 nM T56367 CV04DH 21920370 IC50 > 101000 nM T56367 CRO37P 44274658 IC50 = 75000 nM T56367 C35KNC 44274717 IC50 = 97000 nM T56367 CU36PK 44274868 IC50 > 100000 nM T56367 CDN62V 44274869 IC50 = 430 nM T56367 CA6J8T 44274920 IC50 = 18000 nM T56367 C7NHE8 44279839 IC50 = 380000 nM T56367 COBW92 44301890 IC50 = 39000 nM T56367 C8A2JP 44311854 IC50 = 40000 nM T56367 C5SBO6 44311855 IC50 = 8400 nM T56367 CL80RT 44314758 IC50 = 19000 nM T56367 C7VBP1 44314851 IC50 = 22000 nM T56367 C47XKT 44314914 IC50 = 25000 nM T56367 C3ID9H 44314916 IC50 > 100000 nM T56367 CAF5L9 44314918 IC50 = 45000 nM T56367 CWSU53 44314924 IC50 = 41000 nM T56367 C9YQ2M 44314926 IC50 = 12000 nM T56367 CD3V8J 44314928 IC50 = 20000 nM T56367 CW3P2M 44315107 IC50 > 100000 nM T56367 CC6F4N 44315110 IC50 = 20000 nM T56367 CZ16IY 44324251 IC50 > 100000 nM T56367 CCX9Z3 44324252 IC50 > 100000 nM T56367 CG6UT1 44324296 IC50 > 100000 nM T56367 C8M4WJ 44324373 IC50 > 100000 nM T56367 CY5HZ7 44324390 IC50 > 100000 nM T56367 C5KYV6 44324391 IC50 > 100000 nM T56367 C5C4QX 44324507 IC50 > 100000 nM T56367 CCOZ32 44339609 IC50 = 149000 nM T56367 C6EBY9 44367306 Ki = 16000 nM T56367 C7MI2E 44367386 IC50 > 1000000 nM T56367 CT8NH9 44383851 IC50 > 10000 nM T56367 C19CRH 44383901 IC50 = 2500 nM T56367 CR9O3I 44383902 IC50 = 450 nM T56367 CW47HV 44383906 IC50 = 1150 nM T56367 CL86MY 44383907 IC50 > 10000 nM T56367 CW63HQ 44383912 IC50 > 10000 nM T56367 CF98LG 44384286 IC50 > 10000 nM T56367 CN1WS7 44384345 IC50 > 30000 nM T56367 C01XPL 44384404 IC50 = 3500 nM T56367 CWPR87 44384405 IC50 = 770 nM T56367 C59SDR 44384406 IC50 = 1600 nM T56367 C7WT4G 44384540 IC50 = 1800 nM T56367 C4RQB0 44384541 IC50 = 1820 nM T56367 CRZ5G8 44384546 IC50 = 3100 nM T56367 C6W4GY 44384713 IC50 = 4000 nM T56367 CKH7M8 44384714 IC50 = 4600 nM T56367 C0ZGU6 44385109 IC50 = 910 nM T56367 CE80VB 44385244 IC50 = 1020 nM T56367 CH5GU8 44385282 IC50 = 650 nM T56367 CL50UE 44385283 IC50 = 1220 nM T56367 CQ0S7E 44386000 IC50 = 36000 nM T56367 CHDN54 44386045 IC50 = 20000 nM T56367 CBT82J 44386129 IC50 = 36000 nM T56367 CV1F8W 44386133 IC50 = 4900 nM T56367 CP37LE 44386323 IC50 > 25000 nM T56367 C69DVN 44386324 IC50 = 41000 nM T56367 CWE39G 44386327 IC50 = 1200 nM T56367 CL7OS2 44386388 IC50 = 19000 nM T56367 C2RTX1 44386433 IC50 > 50000 nM T56367 CPQC46 44386434 IC50 = 15000 nM T56367 CD8VL7 44387049 IC50 > 25000 nM T56367 CC9HR5 44387117 IC50 = 54000 nM T56367 C13HPW 44393651 IC50 = 20100 nM T56367 CJ6GB5 44393709 IC50 = 1280 nM T56367 CQP01D 44393950 IC50 = 28840 nM T56367 CU1CQ8 44394047 IC50 = 2980 nM T56367 CJYC83 44397324 IC50 > 10000 nM T56367 CZUY06 44397327 IC50 > 10000 nM T56367 CB64FY 44397328 IC50 = 1810 nM T56367 CDJ87T 44397345 IC50 > 10000 nM T56367 C5CTF6 44397346 IC50 = 8000 nM T56367 CU3BF4 44397365 IC50 > 10000 nM T56367 C4VS1H 44397382 IC50 = 2700 nM T56367 CQD8Z7 44397386 IC50 = 2410 nM T56367 CCL9D6 44397387 IC50 = 3940 nM T56367 C7MZ8J 44397413 IC50 > 10000 nM T56367 CF2AP3 44397474 IC50 = 5700 nM T56367 C6FJV7 44397494 IC50 = 2800 nM T56367 CU13ES 44397515 IC50 = 2000 nM T56367 CTAI27 44397548 IC50 > 10000 nM T56367 CMC12S 44397573 IC50 > 10000 nM T56367 CL15YW 44397574 IC50 > 10000 nM T56367 C6GIS2 44397576 IC50 > 10000 nM T56367 C65PLD 44397577 IC50 > 10000 nM T56367 C3PN4D 44397598 IC50 = 380 nM T56367 CY0KB5 44397600 IC50 > 10000 nM T56367 C86IAQ 44397602 IC50 = 4500 nM T56367 CG2XI7 44397621 IC50 > 10000 nM T56367 C1HBU8 44397622 IC50 > 10000 nM T56367 C1FJH9 44397640 IC50 = 43 nM T56367 CV2Q1K 44397643 IC50 = 1100 nM T56367 CV2M0A 44397708 IC50 > 10000 nM T56367 C8MZF1 44397709 IC50 > 10000 nM T56367 CF1D0Y 44397712 IC50 = 6350 nM T56367 CJIK26 44397727 IC50 = 2670 nM T56367 C2PJ6R 44397748 IC50 > 10000 nM T56367 CAQD83 44397749 IC50 = 1000 nM T56367 C5GLC2 44397761 IC50 > 10000 nM T56367 CQCN29 44397781 IC50 > 10000 nM T56367 C0B2YM 44397782 IC50 = 1360 nM T56367 CWL0A9 44397785 IC50 = 1720 nM T56367 CSN79W 44397799 IC50 > 10000 nM T56367 C20BLM 44397801 IC50 > 10000 nM T56367 CJG87Q 44397802 IC50 = 390 nM T56367 CZF29N 44397816 IC50 = 920 nM T56367 CIVF18 44397836 IC50 = 630 nM T56367 CP18FI 44397837 IC50 > 10000 nM T56367 CRMN86 44397859 IC50 = 7100 nM T56367 C01CAI 44397871 IC50 > 10000 nM T56367 CJ6B1W 44397876 IC50 = 3900 nM T56367 C28ERI 44397877 IC50 = 2930 nM T56367 C6Y9XN 44397888 IC50 = 670 nM T56367 CIOM21 44397889 IC50 = 1720 nM T56367 CX3M5J 44397892 IC50 = 200 nM T56367 CVB7K2 44397908 IC50 > 10000 nM T56367 CP8CW5 44397940 IC50 > 10000 nM T56367 CFHR09 44397941 IC50 > 10000 nM T56367 CP62TK 44397956 IC50 = 4480 nM T56367 C6UY9Z 44397957 IC50 > 10000 nM T56367 C23GTH 44397958 IC50 = 3870 nM T56367 CG36QI 44397976 IC50 > 10000 nM T56367 CDK84C 44397977 IC50 > 10000 nM T56367 CW65CR 44397987 IC50 > 10000 nM T56367 C1DQW5 44397991 IC50 = 4520 nM T56367 CP8F9A 44397992 IC50 > 10000 nM T56367 CI1F5C 46239840 Ki >= 770 nM T56367 C26XVS 46240044 Ki >= 4793 nM T56367 CE4JU7 46842025 IC50 > 10000 nM T56367 CR8JC2 46842169 IC50 > 10000 nM T56367 CZS03D 50902030 Ki > 4274 nM T56367 CH2Z1E 50902289 Ki > 7100 nM T56367 C4HJL2 50902291 Ki > 7950 nM T56367 C6A1IU 50902549 Ki > 2000 nM T56367 C3Y2AV 50903255 Ki > 2000 nM T56367 C6C8RD 66802145 IC50 = 2350 nM T56367 CF03DW 90168772 IC50 > 20000 nM T56367 CM6J9K 90168778 IC50 > 20000 nM T56367 CVYK24 118556943 IC50 > 50000 nM T56367 C1QMI8 135401477 IC50 = 790 nM T56367 C17YXR 135406983 IC50 = 300 nM T56367 C1Z3WH 135430893 IC50 = 1000 nM T56367 CAJU63 135430952 IC50 = 50 nM T56367 CZJY69 135442775 IC50 > 100000 nM T56367 C0IE4A 135443738 IC50 = 1000 nM T56367 CQW8U9 135456038 IC50 = 10 nM T56367 C0BQH8 135456061 IC50 = 30 nM T56367 CR6B9J 135456675 IC50 > 100000 nM T56367 CTN73W 135467948 IC50 = 10 nM T56367 CHSI34 135469671 IC50 = 30 nM T56367 CADL53 135475879 IC50 = 200 nM T56367 CJS37E 135482260 IC50 = 610 nM T56367 CUNL35 135484025 IC50 = 1000 nM T56367 CEZ5P3 135487732 IC50 = 20 nM T56367 CHO1Z5 135489408 IC50 > 1000 nM T56367 CP71WA 135528334 IC50 > 100000 nM T56367 C8E3OA 135531470 IC50 > 100000 nM T56367 CM3GD7 135532874 IC50 = 500 nM T56367 C4ASW0 135544141 IC50 = 300 nM T56367 CYE4C5 135544159 IC50 > 1000 nM T56367 C7M1TE 135604959 IC50 = 30 nM T56367 C6I3HM 135678134 IC50 = 200 nM T56367 CCB89G 135723513 IC50 = 40 nM T56367 CTE50H 135757341 IC50 = 10 nM T56367 CG1AN3 135790070 IC50 = 50 nM T56367 C3PO9K 135856789 IC50 = 3560 nM T56367 C9UK1F 136132272 IC50 = 1000 nM T56367 CBO5H3 136132273 IC50 = 500 nM T56367 CPY6I0 136132274 IC50 = 800 nM T56367 C4ZBT6 136132277 IC50 = 1000 nM T56367 CJ9QG1 136132278 IC50 = 10 nM T56367 C23BTX 136132279 IC50 > 1000 nM T56367 C1BFD5 136132280 IC50 > 1000 nM T56367 CQW7T0 136197286 IC50 = 3640 nM T56367 C2DA1W 155561694 IC50 > 500000 nM T56367 CQ2R0W 155568588 IC50 > 500000 nM T56367 D00YPO 14032753 IC50 = 75000 nM T56367 D0I6XA 149784 Ki > 200000 nM T56367 D0J0CB 2753 Ki = 22000 nM T56367 D0LZ5R 5368 IC50 > 100000 nM T56367 D0R6MT 3758 IC50 = 3400 nM T56367 D0RC4F 72103 IC50 = 16000 nM T56367 D0V4WB 149790 IC50 > 16000 nM T44068 D01UXC 2249 IC50 = 1.77 nM T44068 D03DJL 6918554 Ki = 91 nM T44068 D03GCJ 2583 Ki = 1.9 nM T44068 D03ROX 2369 IC50 = 37.1 nM T44068 D03WEX 9966051 Ki = 46 nM T44068 D04JEE 4946 Ki = 1.4 nM T44068 D04KJO 3410 EC50 = 12.59 nM T44068 D04PHC 5816 EC50 = 290 nM T44068 D04VMT 5253 IC50 = 8900 nM T44068 D05UVD 33624 Ki = 5.37 nM T44068 D0F2PO 4828 Ki = 0.52 nM T44068 D0I2MK 4171 Ki = 55 nM T44068 D0I8FI 3779 EC50 = 0.084 nM T44068 D0L5YV 5152 EC50 = 199.53 nM T44068 D0Y5AM 444031 EC50 = 39.81 nM T44068 D06UKG 9849699 Ki = 0.023 nM T44068 D07WHS 5312115 Ki > 100000 nM T44068 D0A5EF 9887812 Ki = 398.11 nM T44068 D0DH5X 44472635 IC50 > 20000 nM T44068 D0I2XM 3038500 IC50 = 2300 nM T44068 D0LI1C 44469321 IC50 > 10000 nM T44068 D0MT5C 16118894 IC50 = 170 nM T44068 D00OWF 5280953 Ki > 10000 nM T44068 D01SWK 5493324 EC50 = 6.4 nM T44068 D01VAB 2119 Ki = 2.818 nM T44068 D02KMG 9892481 EC50 = 25.12 nM T44068 D04YJU 9829836 IC50 = 200 nM T44068 D0C5PA 183812 Ki = 3922 nM T44068 D0L5TJ 10527469 Ki = 10600 nM T44068 D0M7LV 5761 Ki = 140 nM T44068 D0Y1PG 9841972 Ki = 1130 nM T44068 D0ZG9N 132337 IC50 > 10000 nM T44068 C6TQ7E 2685 Ki = 1.2 nM T44068 CYG2P9 2755 EC50 = 7.413 nM T44068 CZUI83 2769 IC50 > 10000 nM T44068 CJQE97 5581 EC50 = 14 nM T44068 C5H9CN 9287 Ki = 3776 nM T44068 CS9N5R 70541 Ki = 537.03 nM T44068 CPI2E4 80447 IC50 = 13000 nM T44068 C7X0FY 81430 IC50 = 8000 nM T44068 CT6MJ0 83111 IC50 = 12000 nM T44068 CDOJ58 83113 IC50 = 38000 nM T44068 CB6G3Z 91536 Ki = 1.4 nM T44068 C38YOB 91965 IC50 = 14000 nM T44068 C7IPU1 93601 Ki = 213.8 nM T44068 C7D1MY 97269 IC50 > 100000 nM T44068 C3JXH7 97478 IC50 = 15000 nM T44068 CH20FW 121848 IC50 = 37.9 nM T44068 CKP25M 121881 Ki < 1000 nM T44068 CZC0Q1 130400 IC50 = 2400 nM T44068 C3CQK6 131847 IC50 = 160 nM T44068 CZL87W 133999 IC50 > 10000 nM T44068 C96ASF 164451 Ki = 300 nM T44068 CLK7P3 169713 IC50 > 10000 nM T44068 C8WG7P 203685 Ki = 64.57 nM T44068 C0MOL1 204665 Ki = 1.445 nM T44068 CF10IQ 208932 IC50 = 1600 nM T44068 C9G0KB 213051 EC50 = 14 nM T44068 C39OMI 269722 IC50 = 38000 nM T44068 CPA9F2 443372 EC50 = 7.943 nM T44068 CX75UZ 598754 Ki = 220 nM T44068 CDE4L9 702318 Ki = 1584.89 nM T44068 CG72WR 770558 Ki = 1258.93 nM T44068 C08WCU 851833 Ki = 107.15 nM T44068 CP94RB 2447484 IC50 = 29.4 nM T44068 CV3KM9 2447486 IC50 = 43.3 nM T44068 CDLO23 2723782 Ki = 741.31 nM T44068 CS8N5X 2736067 Ki = 85.11 nM T44068 C7K3GJ 2736205 Ki = 1584.89 nM T44068 C17WFV 2770390 Ki = 293 nM T44068 CP5GF0 2778334 Ki = 2511.89 nM T44068 CRS35B 2796082 Ki > 10000 nM T44068 C9MJD1 3079339 IC50 = 2400 nM T44068 C72IHQ 3207225 Ki = 676.08 nM T44068 CMSB89 3687256 IC50 = 377 nM T44068 C1CK2S 4143663 Ki = 1360 nM T44068 CBC7N9 4276762 Ki = 530 nM T44068 CW2IR6 4421983 Ki = 80 nM T44068 C70GLP 5187268 Ki = 740 nM T44068 CIZ7U3 6603820 Ki = 1500 nM T44068 C3A1FO 6604789 Ki < 10000 nM T44068 C1MW2P 6916441 EC50 = 6.4 nM T44068 C0QRE3 8029710 Ki = 199.53 nM T44068 C7SIU5 9799092 EC50 = 79.43 nM T44068 CGX49B 9800339 EC50 = 358 nM T44068 CH6PX1 9801145 EC50 = 5011.87 nM T44068 C7ZQ3D 9803765 EC50 = 48700 nM T44068 C68VZH 9803988 EC50 > 3200 nM T44068 CRJ79X 9804536 EC50 = 14.79 nM T44068 CE0DI5 9804612 Ki < 1000 nM T44068 CUY3S0 9810596 IC50 = 2300 nM T44068 C7HQ9N 9816183 Ki = 60.6 nM T44068 CM48YW 9821129 Ki = 1300 nM T44068 CD7TA2 9823696 EC50 = 794.33 nM T44068 CD2U3O 9826638 IC50 = 1800 nM T44068 CB6O2M 9827999 Ki = 9490 nM T44068 CYR8O6 9831168 EC50 = 19 nM T44068 CK7WI5 9832011 IC50 = 2000 nM T44068 CK7DS2 9842600 EC50 = 1500 nM T44068 C3JYI0 9845280 EC50 = 1258.93 nM T44068 C1CEO4 9845282 EC50 = 6.31 nM T44068 C0OS8W 9847067 EC50 = 39.81 nM T44068 CY3DL8 9849126 EC50 = 25.12 nM T44068 C9FAP3 9853471 EC50 = 1800 nM T44068 CB6R3T 9858463 Ki = 200 nM T44068 CZY34F 9860739 Ki = 2.37 nM T44068 CBD6E0 9866060 Ki = 227 nM T44068 CFVG52 9866061 Ki > 10000 nM T44068 CJIR63 9871386 EC50 = 7.943 nM T44068 CJ72CL 9871525 IC50 = 230 nM T44068 C1L6XP 9871887 Ki = 2.042 nM T44068 C51FVW 9872550 EC50 > 3160 nM T44068 CVF5O3 9873245 IC50 = 27 nM T44068 CSRF54 9873257 EC50 = 1900 nM T44068 CA43HC 9874175 EC50 > 10000 nM T44068 CDQ84R 9888047 EC50 = 100 nM T44068 C5L3VF 9893058 EC50 = 50.12 nM T44068 CRV61G 9896742 EC50 = 3 nM T44068 CMC06V 9896817 EC50 = 970 nM T44068 CYWQ50 9906447 Ki > 10000 nM T44068 C6CZ3G 9906777 IC50 > 10000 nM T44068 CQP6X3 9906822 EC50 = 0.13 nM T44068 CUHF02 9908924 Ki = 7600 nM T44068 C2A1CZ 9912443 EC50 > 1000 nM T44068 CMH72E 9912580 IC50 = 110 nM T44068 CDH69A 9915235 EC50 > 100000 nM T44068 CYH07G 9915238 IC50 = 8000 nM T44068 CH9OT6 9917962 EC50 = 41 nM T44068 CW7YJ1 9924779 Ki = 270 nM T44068 C1XSL4 9927453 EC50 = 1.9 nM T44068 C92XMC 9933039 EC50 = 210 nM T44068 CYVZ47 9934284 Ki = 794.33 nM T44068 C7MO0Z 9938030 IC50 = 3000 nM T44068 CZM1E2 9946573 Ki = 400 nM T44068 C9PVT1 9947512 Ki = 37 nM T44068 CCN27K 9958539 EC50 = 2 nM T44068 CM6I4O 9960584 Ki = 2600 nM T44068 CCA49K 9962058 EC50 > 1000 nM T44068 CB3AQ9 9967732 Ki = 400 nM T44068 CY78ZQ 9982903 Ki = 7.8 nM T44068 CFTV18 9984028 EC50 < 5011.87 nM T44068 C1NYC0 10002049 EC50 > 1000 nM T44068 CEF4Y3 10003858 EC50 = 500 nM T44068 CO3DB4 10007337 IC50 = 5500 nM T44068 CP0H1B 10008017 EC50 = 60 nM T44068 C2EUY0 10035109 Ki > 10000 nM T44068 CTE2I9 10048077 EC50 = 250 nM T44068 CFBU26 10049403 Ki = 15 nM T44068 CJP10L 10051943 Ki = 181.97 nM T44068 CWJ25B 10054165 IC50 = 2400 nM T44068 CRU28L 10054896 IC50 = 1290 nM T44068 CBVG28 10075383 EC50 = 340 nM T44068 C1SXV8 10075766 Ki = 1.4 nM T44068 CVE2T1 10076176 EC50 = 501.19 nM T44068 C8TBK0 10076548 EC50 = 40 nM T44068 C7SL6M 10076885 IC50 = 8333 nM T44068 CP7WF3 10092953 EC50 = 63 nM T44068 CSNP15 10099346 IC50 = 4800 nM T44068 CL81PN 10099459 IC50 = 5000 nM T44068 CRK6B0 10101116 IC50 = 8400 nM T44068 CP6L3C 10112732 IC50 = 590 nM T44068 CA4MV1 10112744 Ki = 97 nM T44068 C8SAN2 10113837 EC50 = 20 nM T44068 CQW48U 10117815 Ki > 10000 nM T44068 CJ31XM 10119061 IC50 = 730 nM T44068 CLB01Q 10119515 EC50 = 260 nM T44068 C07WRX 10121328 EC50 = 1000 nM T44068 CIX83H 10131985 Ki = 170 nM T44068 CCRO89 10132882 Ki = 100 nM T44068 CE27RV 10135864 EC50 > 10000 nM T44068 CZ8AQ7 10136220 Ki = 130 nM T44068 C8ZK3L 10138809 IC50 = 480 nM T44068 CZ0J7I 10140092 Ki = 6000 nM T44068 CP0K9U 10140428 EC50 > 100000 nM T44068 CTZ03I 10140889 EC50 = 164 nM T44068 C4B7XL 10140996 Ki = 3200 nM T44068 C0FS3J 10142284 EC50 = 85 nM T44068 CO3F6S 10144004 EC50 > 100000 nM T44068 CD0RL9 10145446 EC50 = 2050 nM T44068 CHZQ30 10145482 EC50 = 1010 nM T44068 CDHS42 10155942 Ki = 210 nM T44068 CCP74I 10160281 EC50 > 1000 nM T44068 C27MZY 10160636 IC50 = 980 nM T44068 CGJ10H 10162297 Ki = 3600 nM T44068 CMK05F 10180590 EC50 = 251.19 nM T44068 CB9HW6 10187201 EC50 = 610 nM T44068 C8EOD0 10187653 EC50 = 489 nM T44068 CZHJ01 10189730 EC50 = 423 nM T44068 C1H8AB 10201549 Ki = 100 nM T44068 C4YW9V 10202462 EC50 = 251.19 nM T44068 CCO4D7 10202842 EC50 = 511 nM T44068 C56USA 10203169 EC50 = 19.95 nM T44068 C6Y5JB 10205362 IC50 = 290 nM T44068 C9N1WB 10205463 EC50 = 943 nM T44068 CF5RL8 10206782 IC50 = 240 nM T44068 C2MX7I 10207208 Ki = 560 nM T44068 C1H0JA 10207209 Ki = 47000 nM T44068 C3A2UK 10209243 EC50 > 10000 nM T44068 C2KEW4 10209574 EC50 = 522 nM T44068 CF6R2U 10217757 EC50 = 10 nM T44068 CPE8M6 10225563 EC50 = 7.943 nM T44068 C2I6BY 10227108 Ki > 10000 nM T44068 C4KTP1 10231394 EC50 = 10900 nM T44068 C9Y4AT 10231679 Ki = 690 nM T44068 CF4Z1B 10232096 EC50 = 254 nM T44068 CV4QB7 10232593 EC50 = 88 nM T44068 C2YDG7 10233153 EC50 = 50 nM T44068 CO64WJ 10236758 Ki = 47863.01 nM T44068 CSC3V2 10238776 EC50 = 63.1 nM T44068 CDCP62 10239722 EC50 = 2.512 nM T44068 CYBX59 10258518 IC50 = 2500 nM T44068 C1KR8D 10273469 Ki = 150 nM T44068 CBFQ89 10275157 EC50 = 350 nM T44068 CV25SE 10278987 EC50 > 100000 nM T44068 C1EZ4U 10280301 EC50 = 109 nM T44068 C6YUK7 10281165 EC50 = 1015 nM T44068 C9TLW7 10282871 IC50 = 16 nM T44068 CO24KP 10283146 EC50 = 30 nM T44068 CF4Y7P 10283539 EC50 = 353 nM T44068 C9S2EY 10287658 Ki = 31622.78 nM T44068 C5TEI1 10288976 EC50 = 39.81 nM T44068 C7F6LZ 10291064 Ki = 140 nM T44068 CD1S6J 10292413 Ki = 360 nM T44068 CV42BX 10297331 Ki = 50 nM T44068 CIW29S 10298567 EC50 = 4 nM T44068 C2FSP4 10301101 EC50 = 100000 nM T44068 C3RP8X 10301445 EC50 > 1000 nM T44068 CUJ3M7 10302342 EC50 = 187 nM T44068 C1U3DW 10302915 EC50 = 750 nM T44068 C9PK4A 10304565 EC50 = 525 nM T44068 COES23 10304786 EC50 > 1000 nM T44068 CUML26 10305108 EC50 = 390 nM T44068 C42ZDS 10310047 Ki = 31622.78 nM T44068 COL3N7 10310564 Ki = 12589.25 nM T44068 CLO20K 10311070 Ki = 19952.62 nM T44068 C3E5CB 10337773 Ki < 100000 nM T44068 C1PSZ4 10346448 EC50 = 630.96 nM T44068 CZ26AE 10347866 IC50 = 18000 nM T44068 C7H9PZ 10371216 IC50 = 2300 nM T44068 CDRL02 10393774 EC50 = 2000 nM T44068 CA2N8B 10406968 Ki = 28 nM T44068 C5QI3T 10416448 IC50 = 20000 nM T44068 C6URQ9 10416656 IC50 = 1200 nM T44068 C38QCR 10431900 Ki = 2300 nM T44068 CB9U6O 10436455 Ki = 140 nM T44068 C6ZIY2 10437614 IC50 = 1000 nM T44068 C59OLP 10438390 IC50 = 2000 nM T44068 C8W4IC 10457669 Ki = 31 nM T44068 CXCL36 10459124 Ki = 160 nM T44068 COV85C 10472143 Ki = 76 nM T44068 CA20IB 10483845 IC50 = 21000 nM T44068 CQKI17 10544781 Ki = 6165.95 nM T44068 CQ4Z8H 10553602 EC50 = 50 nM T44068 CL0MJ3 10553603 EC50 = 100 nM T44068 CK87QN 10575455 EC50 = 1200 nM T44068 CB83SX 10601234 EC50 = 1600 nM T44068 C4NWL1 10602703 EC50 > 10000 nM T44068 CW2S8I 10626150 EC50 = 4500 nM T44068 CWP9M1 10627736 IC50 = 1800 nM T44068 C51DIX 10648298 EC50 = 9800 nM T44068 CX9WA0 10651078 IC50 = 2600 nM T44068 C1C6KV 10651147 EC50 = 43700 nM T44068 C8WX4M 10722793 EC50 = 2700 nM T44068 C6R5QN 10745501 EC50 > 1000 nM T44068 CFJA38 10746499 IC50 = 1900 nM T44068 CQA4E2 10841171 IC50 = 2500 nM T44068 CHM6J4 10841426 IC50 = 2000 nM T44068 C05CGB 10863093 EC50 = 100 nM T44068 C92OSW 10902809 EC50 = 5.012 nM T44068 CY1QM6 10940242 EC50 = 794.33 nM T44068 CNB39C 10947658 Ki = 400 nM T44068 CC6V1Z 11002571 EC50 = 630.96 nM T44068 CRJ5L3 11003341 EC50 = 251.19 nM T44068 C8V7XF 11005613 EC50 = 19.95 nM T44068 C6TAO1 11026016 EC50 = 5.012 nM T44068 CCKZ08 11038599 EC50 = 398.11 nM T44068 CZI9B1 11060184 EC50 = 794.33 nM T44068 C23NHX 11091850 EC50 = 25.12 nM T44068 C2N0BD 11124502 EC50 < 794.33 nM T44068 C8FVK0 11134054 EC50 = 3.162 nM T44068 C41RIK 11152564 EC50 = 130 nM T44068 C62GDB 11156916 EC50 > 1000 nM T44068 C34JRO 11169365 EC50 = 6.31 nM T44068 C6CL1Y 11178830 Ki = 1258.93 nM T44068 CY04IB 11180293 EC50 = 10 nM T44068 CQS49K 11188590 Ki = 133 nM T44068 COE80P 11189433 EC50 = 711.5 nM T44068 CS5G0X 11218492 Ki = 2344.23 nM T44068 CUGE45 11224220 EC50 = 300 nM T44068 CB69KG 11224275 EC50 = 690 nM T44068 CX6EI1 11235459 EC50 > 1000 nM T44068 C90WSG 11248705 Ki = 398.11 nM T44068 CD2VF8 11268355 EC50 = 0.13 nM T44068 CNJZ06 11270069 EC50 = 9.4 nM T44068 CBJ49T 11270071 EC50 = 47 nM T44068 CRFS12 11272641 EC50 = 800 nM T44068 CJS9C0 11304851 IC50 > 25000 nM T44068 CQ08YH 11340895 EC50 > 1000 nM T44068 CGQ2D0 11342656 IC50 = 2500 nM T44068 CUNJ91 11352782 EC50 > 1000 nM T44068 C0MG9U 11381882 EC50 = 140 nM T44068 C0YB8T 11398536 EC50 = 900 nM T44068 CMX29E 11420551 EC50 = 260 nM T44068 C85LYP 11430418 IC50 > 1000 nM T44068 CQC36P 11432806 EC50 = 18 nM T44068 CL1M5W 11453340 EC50 > 1000 nM T44068 C6TA1B 11476004 EC50 = 780 nM T44068 CW3YR2 11495581 EC50 = 794.33 nM T44068 C16TWK 11508052 IC50 > 10000 nM T44068 CXWO08 11522273 IC50 > 10000 nM T44068 CAT27M 11523842 IC50 = 0.11 nM T44068 CV6IN9 11539348 EC50 = 103.4 nM T44068 C5PQR9 11546170 IC50 = 0.08 nM T44068 CZ62AI 11546349 EC50 = 794.33 nM T44068 CAWR47 11556330 IC50 = 3300 nM T44068 CWGO05 11567751 EC50 = 101 nM T44068 CWM5K6 11575154 EC50 = 10000 nM T44068 CP2WJ8 11592062 EC50 = 3.981 nM T44068 CY15EM 11605652 EC50 = 5011.87 nM T44068 C8A7SC 11617407 Ki = 1.8 nM T44068 C12YSL 11625333 Ki = 421 nM T44068 C74VKM 11625493 EC50 = 200 nM T44068 CAU8C5 11625619 Ki = 1.9 nM T44068 CKZ65X 11632691 EC50 = 207 nM T44068 CMIC92 11647002 Ki = 70 nM T44068 C7ZTC8 11647543 EC50 = 630.96 nM T44068 C1J4XV 11661536 EC50 = 3162.28 nM T44068 C1W6ZT 11668125 EC50 = 215 nM T44068 COHD32 11669967 EC50 = 2511.89 nM T44068 CKJU26 11703823 EC50 = 171 nM T44068 CD31TA 11718543 EC50 = 5011.87 nM T44068 CPG15O 11743399 IC50 > 1000 nM T44068 CU5I1X 11757304 Ki = 5.2 nM T44068 CT1OL3 11758172 EC50 = 2600 nM T44068 C4ISZ7 11810896 EC50 = 7.943 nM T44068 CN9M8E 11811722 IC50 = 3590 nM T44068 C8JQL7 11957735 IC50 > 10000 nM T44068 C3BXJ2 12017001 IC50 = 3000 nM T44068 CF5TK1 12017002 IC50 = 6500 nM T44068 C38DZJ 12017003 IC50 = 31000 nM T44068 CN5A2D 12017004 IC50 = 7500 nM T44068 C40KFM 12017005 IC50 = 2000 nM T44068 C0G3XR 12017006 IC50 = 2100 nM T44068 C2FZ3H 12017007 IC50 = 1900 nM T44068 CDZQ57 12017010 IC50 = 4700 nM T44068 CEC98K 12017011 IC50 = 2400 nM T44068 C02SVL 12017012 IC50 = 1200 nM T44068 C1ZH0K 12017013 IC50 = 6500 nM T44068 C31JDV 12017014 IC50 = 2000 nM T44068 CLIX97 12017015 IC50 = 8000 nM T44068 CO0ST4 12017016 IC50 = 1000 nM T44068 C7Z8WC 12017017 IC50 = 6500 nM T44068 C60OVP 12017018 IC50 = 42000 nM T44068 CPU75A 12043155 IC50 = 26000 nM T44068 C1MFE0 12043156 IC50 = 5500 nM T44068 CR0T9I 12043157 IC50 = 1970 nM T44068 C4U9KY 12043158 IC50 = 10000 nM T44068 CW0XL2 12043159 IC50 = 70000 nM T44068 C7I2CM 12049914 IC50 = 8700 nM T44068 C5M8FQ 12049915 IC50 = 40000 nM T44068 C49XHR 12049916 IC50 = 2600 nM T44068 C7TAQ6 12049917 IC50 = 5600 nM T44068 CDI75Z 12049918 IC50 = 1300 nM T44068 C0LF7J 12049919 IC50 = 3000 nM T44068 C6JWS8 12049920 IC50 = 2500 nM T44068 CU7A5R 12049921 IC50 = 28000 nM T44068 CDZF95 12049922 IC50 = 2600 nM T44068 CZ4V2K 12049923 IC50 = 10000 nM T44068 C8DUY7 12049924 IC50 = 930 nM T44068 CF0IG7 12049925 IC50 = 920 nM T44068 C3U1SP 12049926 IC50 = 6200 nM T44068 CO8BW3 13208878 IC50 = 234.42 nM T44068 CZI4G6 13208884 IC50 = 97.72 nM T44068 C03EXV 13345218 EC50 = 0.9 nM T44068 CDI64R 14664343 IC50 = 2800 nM T44068 CW2CX6 14664345 IC50 = 21000 nM T44068 CCR3Y1 14664347 IC50 = 18000 nM T44068 C0Q6KE 14664348 IC50 = 2600 nM T44068 CI1L9P 14739889 IC50 = 2400 nM T44068 C25HZI 14739891 IC50 = 7300 nM T44068 CV8D7G 14739892 IC50 = 800 nM T44068 C0M1UP 14739893 IC50 = 33100 nM T44068 CIR0Q4 14739897 IC50 = 19200 nM T44068 C1R5FU 14739901 IC50 = 3300 nM T44068 CBQT63 14739905 IC50 = 40 nM T44068 C8NO3D 14739906 IC50 = 270 nM T44068 CD4JZ0 14739907 IC50 = 270 nM T44068 CE5LK3 14739908 IC50 = 5100 nM T44068 CFC0D6 14823035 Ki = 170 nM T44068 CMO81H 14925759 Ki = 32359.37 nM T44068 C10CRK 14998846 IC50 = 3000 nM T44068 CMU79D 14998847 IC50 = 31000 nM T44068 C95XQS 14998848 IC50 = 540 nM T44068 C2FHB7 14998849 IC50 = 1700 nM T44068 CGP94Z 14998850 IC50 = 230 nM T44068 CM3Q9V 14998851 IC50 = 3300 nM T44068 C39CAP 14998852 IC50 = 2300 nM T44068 C1BUN5 14998853 IC50 = 26000 nM T44068 CAG7Y3 14998855 IC50 = 1100 nM T44068 CNX73O 14998858 IC50 = 1100 nM T44068 CI16HW 15077948 Ki = 7.4 nM T44068 C0BQ4X 15077955 Ki = 300 nM T44068 C1UK2H 15077956 Ki = 820 nM T44068 CZB1M6 15123375 IC50 = 680 nM T44068 CVHW24 15123377 IC50 > 100000 nM T44068 CKFL78 15221053 Ki = 3440 nM T44068 C9HLK1 15221055 Ki = 58100 nM T44068 C25CVZ 15483879 IC50 = 8000 nM T44068 CLNE19 15483880 IC50 = 5000 nM T44068 CUK85J 15483883 IC50 = 4000 nM T44068 CSDO83 15523859 IC50 = 580 nM T44068 C6Q9FZ 15523860 IC50 = 8500 nM T44068 CKP61A 15523861 IC50 = 4000 nM T44068 C1VWH5 15580747 Ki = 2400 nM T44068 CCTM64 16049024 IC50 = 7.943 nM T44068 C17ZSM 16049026 IC50 = 3.162 nM T44068 CC3O5H 16049028 EC50 = 3.981 nM T44068 C71EWF 16049029 IC50 = 3.162 nM T44068 C3OC9G 16049087 IC50 = 7.943 nM T44068 CD41WM 16049088 IC50 = 7.943 nM T44068 C63MIJ 16049090 IC50 = 251.19 nM T44068 C8B4VS 16049158 IC50 = 50.12 nM T44068 CE85LR 16049160 IC50 = 125.89 nM T44068 C27VPK 16049162 IC50 = 100 nM T44068 C6Z4CS 16049234 EC50 = 100 nM T44068 CP06JS 16049309 EC50 = 39.81 nM T44068 CB3MN6 16049374 EC50 = 100 nM T44068 C4QJE9 16049376 EC50 = 63.1 nM T44068 C19EUK 16049377 EC50 = 31.62 nM T44068 CKY42H 16049448 EC50 = 100 nM T44068 CC4F0L 16049450 EC50 = 100 nM T44068 CH8KY4 16126657 EC50 > 10000 nM T44068 C42ELY 16219010 EC50 < 794.33 nM T44068 CERP08 16219807 Ki < 10000 nM T44068 C9JE3V 16222317 EC50 > 1000 nM T44068 CDV38P 16222840 EC50 = 110 nM T44068 C9ONT1 16222940 EC50 = 150 nM T44068 C3C9WR 16223045 EC50 > 1000 nM T44068 CHJ65G 16223251 EC50 = 12 nM T44068 CZ2IS9 16660294 Ki > 10000 nM T44068 C2P0SB 16717791 Ki = 478 nM T44068 CHRG71 16738927 IC50 > 794.33 nM T44068 C3T5HF 21509921 Ki > 10000 nM T44068 C1JBM4 22063464 EC50 = 42 nM T44068 C72IMX 22171479 EC50 = 63 nM T44068 C7PQ8B 22171507 EC50 = 9.2 nM T44068 CCMB98 22171637 EC50 = 37 nM T44068 CN9Z2S 23661589 EC50 = 1258.93 nM T44068 CWEM23 24321330 Ki = 250 nM T44068 CC9G6L 24733400 Ki = 251.19 nM T44068 C1V2UI 24764458 EC50 > 10000 nM T44068 C7QK6D 24804878 EC50 = 86 nM T44068 CRV58X 24822304 EC50 = 1.4 nM T44068 CST3O6 24822310 EC50 = 280 nM T44068 C3C7SF 24822313 EC50 > 100 nM T44068 CTJD72 24822469 EC50 = 200 nM T44068 CIWN92 24822472 EC50 = 570 nM T44068 C8F7MR 24822643 EC50 = 20 nM T44068 C86IOK 24822645 EC50 = 30 nM T44068 CN4H3E 24822648 EC50 = 18 nM T44068 C4H6MR 24822815 EC50 = 350 nM T44068 CV1FP0 24822817 EC50 = 55 nM T44068 CBRX49 24822819 EC50 > 1000 nM T44068 CG13QX 24822970 EC50 = 300 nM T44068 CL4WP6 24822971 EC50 = 3.1 nM T44068 CWAO15 24822972 EC50 = 6.5 nM T44068 CVH1N4 24822974 EC50 > 1000 nM T44068 CBS82N 24823127 EC50 = 720 nM T44068 C5NYS2 24823130 EC50 = 380 nM T44068 C0Q2ZB 24823131 EC50 = 260 nM T44068 CU3D5Q 24823134 EC50 > 1000 nM T44068 C7US9I 24823292 EC50 > 1000 nM T44068 CHUC65 24823294 EC50 = 260 nM T44068 CCF7Z8 24823296 EC50 = 980 nM T44068 C9MBA4 24823462 EC50 > 1000 nM T44068 CHDE90 24823464 EC50 = 170 nM T44068 CJ9GR6 24823468 EC50 > 100 nM T44068 C5MS2U 24823470 EC50 > 100 nM T44068 CZ7UX0 24823624 EC50 = 3.9 nM T44068 CQ7C8J 24823626 EC50 = 36 nM T44068 C8Z3FQ 24823627 EC50 > 1000 nM T44068 CE8N3Y 24823782 EC50 = 11 nM T44068 C0Q2KI 24824226 EC50 = 64 nM T44068 CT9QC7 24824227 EC50 > 100 nM T44068 C7FT4Z 24824228 EC50 > 100 nM T44068 C0EU5V 24824352 EC50 > 100 nM T44068 CR6N2C 24885648 Ki = 159 nM T44068 C1SFL2 24886595 Ki = 268 nM T44068 C08VXN 24893964 EC50 = 480 nM T44068 CV5YU1 24893966 EC50 = 400 nM T44068 CYN9K4 24894127 EC50 > 10000 nM T44068 C3C0KP 24894134 EC50 > 50000 nM T44068 C7FR5U 24894202 EC50 = 28 nM T44068 C9UV7P 24894315 EC50 = 84 nM T44068 C3W2AI 24894317 EC50 = 15 nM T44068 CGR30O 24894319 EC50 = 510 nM T44068 C5TR9W 24894323 EC50 = 11 nM T44068 C8ZG2O 24895192 EC50 = 320 nM T44068 CS1Q4X 24895194 EC50 > 1000 nM T44068 C3Y6LC 24895196 EC50 > 1000 nM T44068 CN1W9Y 24895259 EC50 = 150 nM T44068 C5AD3B 24895261 EC50 = 130 nM T44068 CW8V3F 24895263 EC50 = 39 nM T44068 CYG8J1 24895265 EC50 = 13 nM T44068 CLJ1U9 24895357 EC50 = 37 nM T44068 CULO78 24895359 EC50 = 83 nM T44068 CT7AM8 24895361 EC50 = 86 nM T44068 CA52PH 24895363 EC50 = 130 nM T44068 C76BAX 24895365 EC50 = 280 nM T44068 CF6SM4 24895557 EC50 = 120 nM T44068 CD26KH 24895559 EC50 = 110 nM T44068 C7YEW8 24895561 EC50 = 52 nM T44068 CG1D9Y 24895563 EC50 = 210 nM T44068 CT5HK9 24895565 EC50 = 91 nM T44068 CZ14LI 24895664 EC50 = 180 nM T44068 CE4K2V 24895667 EC50 = 500 nM T44068 CRN05D 24895669 EC50 = 440 nM T44068 C5OKI6 24895671 EC50 > 1000 nM T44068 CIOG69 24895783 EC50 > 1000 nM T44068 CQO97P 24895787 EC50 = 12 nM T44068 CLV98U 24895789 EC50 = 22 nM T44068 C5QLA9 24895791 EC50 = 62 nM T44068 C13JLE 24900426 IC50 = 19.95 nM T44068 C1U9VL 24900685 IC50 = 158.49 nM T44068 CU3F7K 24900689 IC50 = 50.12 nM T44068 CPLO51 24900749 IC50 = 199.53 nM T44068 CX69CF 24900750 IC50 = 10 nM T44068 CE5W9U 24900751 IC50 = 100 nM T44068 CQDR84 24900811 IC50 = 1258.93 nM T44068 CIL8Q7 24900812 IC50 = 79.43 nM T44068 C9YUP8 24900813 IC50 = 6.31 nM T44068 C63ILV 24900872 IC50 = 63.1 nM T44068 CSF3J2 24900874 IC50 = 794.33 nM T44068 C4AT0P 24900937 IC50 = 316.23 nM T44068 C2NR7M 24900942 IC50 = 63.1 nM T44068 CW0QV2 24901141 IC50 = 12.59 nM T44068 CHWE43 24901143 IC50 = 10 nM T44068 C5ZCX4 24901144 IC50 = 63.1 nM T44068 CNP40V 24901209 IC50 = 79.43 nM T44068 C7MGC9 24901210 IC50 = 158.49 nM T44068 CS6BH7 24901211 IC50 = 251.19 nM T44068 C4JB7G 24901283 IC50 = 158.49 nM T44068 CBS0V5 24901284 IC50 = 7.943 nM T44068 C83MAF 24901285 IC50 = 19.95 nM T44068 CVE24O 24901347 IC50 = 398.11 nM T44068 CV5GY0 24901348 IC50 = 398.11 nM T44068 CFZ5D7 24901349 IC50 = 398.11 nM T44068 CCMQ16 24901351 IC50 = 316.23 nM T44068 CGW2U6 24901413 IC50 = 316.23 nM T44068 COY5H0 24901416 IC50 = 1.995 nM T44068 C4BU6R 24936488 EC50 = 65 nM T44068 CH87SX 24936489 Ki = 975 nM T44068 CIR69S 24936491 EC50 = 6.3 nM T44068 C75UCO 24936492 EC50 = 1.8 nM T44068 CRPN83 24936625 Ki = 6710 nM T44068 CT0ND6 24936626 EC50 = 3.5 nM T44068 CFZT09 24936627 Ki = 9330 nM T44068 CH7TO3 24936763 Ki = 2810 nM T44068 CKD63O 24936881 EC50 = 0.57 nM T44068 CTS43M 24936882 Ki = 1049 nM T44068 C38LFU 24936885 Ki = 287 nM T44068 CL91OF 24937013 Ki = 236 nM T44068 C61SKD 24937014 Ki = 1480 nM T44068 CR13DN 24937016 Ki = 5600 nM T44068 CY4KV6 24937137 Ki = 3970 nM T44068 CNP3A6 24937269 EC50 = 70 nM T44068 CZQH42 24937389 Ki = 484 nM T44068 COLT89 24937390 Ki = 560 nM T44068 C2H1AS 24949260 EC50 > 100 nM T44068 CX8N2G 24949262 EC50 > 1000 nM T44068 C6CGT0 24949264 EC50 > 100 nM T44068 C1G4IU 24949414 EC50 > 100 nM T44068 CME8R0 24949416 EC50 > 100 nM T44068 CH6YJ7 24949418 EC50 > 1000 nM T44068 CH0ZA8 24949420 EC50 = 490 nM T44068 CO2IH8 24949564 EC50 = 480 nM T44068 CMIA50 24949566 EC50 = 360 nM T44068 C2IN7M 24949568 EC50 = 340 nM T44068 CK2NO1 24949570 EC50 > 1000 nM T44068 C4R8MP 24949572 EC50 = 140 nM T44068 CNV6F3 24949720 EC50 = 917 nM T44068 C12RTH 24949722 EC50 = 775 nM T44068 CIJ8T1 24949724 EC50 > 1000 nM T44068 CK70NO 24949726 EC50 = 825 nM T44068 CIL04S 24949728 EC50 = 310 nM T44068 C16RWX 24949883 EC50 = 980 nM T44068 CFN26M 24949885 EC50 > 100 nM T44068 C9FWC3 24949887 EC50 > 100 nM T44068 C4Q1NP 24949889 EC50 = 160 nM T44068 CA5Q4V 24949891 EC50 = 70 nM T44068 C1VE2O 24950053 EC50 = 670 nM T44068 CH2R8Z 24950055 EC50 > 1000 nM T44068 C8FY7G 24950057 EC50 > 1000 nM T44068 CL5CM8 24950059 EC50 = 890 nM T44068 C8HMF4 24950061 EC50 > 1000 nM T44068 C5VTD0 24950234 EC50 = 173 nM T44068 CQ80CT 24950236 EC50 = 69 nM T44068 CFZ85T 24950238 EC50 = 330 nM T44068 CJS80L 24950240 EC50 > 100 nM T44068 C3PB6N 24950242 EC50 > 1000 nM T44068 CH2Q3D 24950401 EC50 = 270 nM T44068 CEU3F6 24950403 EC50 > 1000 nM T44068 C2CD3O 24950405 EC50 > 100 nM T44068 CBX0L5 24950407 EC50 > 100 nM T44068 C6JXL4 24950409 EC50 > 1000 nM T44068 CNR3Y4 24950560 EC50 = 620 nM T44068 C0M1XB 24950562 EC50 > 1000 nM T44068 CH9U4B 24950564 EC50 > 1000 nM T44068 CE0WB4 24950566 EC50 > 1000 nM T44068 CMV2K0 24950568 EC50 = 200 nM T44068 CS7U5E 24950570 EC50 = 650 nM T44068 C5ZG2W 24950716 EC50 > 1000 nM T44068 CLF4U7 24950718 EC50 = 800 nM T44068 CY6I9E 25020250 IC50 = 2351 nM T44068 C6FHK9 25071020 EC50 = 810 nM T44068 CA1EJ2 25120700 Ki = 863 nM T44068 C4MRQ0 27842480 Ki = 77 nM T44068 CAD31R 42611263 EC50 = 316.23 nM T44068 C0FE1J 42625511 EC50 = 251.19 nM T44068 C7GK2I 42625513 EC50 = 501.19 nM T44068 CE6IF3 42625515 EC50 = 501.19 nM T44068 C1BE8M 42625517 EC50 = 1000 nM T44068 CL89KJ 42625587 EC50 = 125.89 nM T44068 CQ4O3V 42625588 EC50 = 1000 nM T44068 C9Q0OM 42625741 EC50 = 1258.93 nM T44068 CBN76E 42625743 EC50 = 79432.82 nM T44068 C6P3JN 42625821 EC50 = 630.96 nM T44068 C3JAT7 42625823 EC50 = 100 nM T44068 C4KE6Z 42625897 EC50 = 630.96 nM T44068 C6YR7G 42625898 EC50 = 1258.93 nM T44068 CA2YO5 42639133 EC50 > 1000 nM T44068 CRF79M 42639311 EC50 = 160 nM T44068 CP0D6A 42639314 EC50 = 220 nM T44068 C6I5KU 42639317 EC50 > 1000 nM T44068 C7J1IV 42639487 EC50 > 1000 nM T44068 CN6G7U 42639489 EC50 > 1000 nM T44068 C1ORB7 42639491 EC50 = 840 nM T44068 CAJ05V 42639494 EC50 > 1000 nM T44068 CCX13B 42639652 EC50 = 490 nM T44068 C9YFJ6 42639654 EC50 = 240 nM T44068 CFK5S7 42639656 EC50 > 1000 nM T44068 CK0X9P 42639806 EC50 = 730 nM T44068 C7IL9X 42639808 EC50 = 750 nM T44068 CTHM06 42639810 EC50 > 1000 nM T44068 CTY09A 42639965 EC50 = 370 nM T44068 C97BUG 42639967 EC50 = 130 nM T44068 C4OU1Q 42639969 EC50 = 320 nM T44068 C9QLJ6 42640120 EC50 > 1000 nM T44068 C21SKJ 42640122 EC50 > 1000 nM T44068 CB4Q8W 44126931 EC50 = 180 nM T44068 CWGQ16 44126933 EC50 = 150 nM T44068 CU8M4H 44127048 EC50 = 590 nM T44068 CXM3V6 44127050 EC50 = 720 nM T44068 CS0B5Z 44127052 EC50 = 960 nM T44068 C4H9TJ 44127054 EC50 = 280 nM T44068 C2IC7Q 44127056 EC50 = 490 nM T44068 CAW50P 44127167 EC50 = 910 nM T44068 CJ0S7Q 44127169 EC50 > 100000 nM T44068 C53MWL 44127171 EC50 = 290 nM T44068 CX2VJ3 44127374 EC50 = 260 nM T44068 C8BRZ2 44127478 EC50 = 660 nM T44068 C6XMJ7 44127479 EC50 = 83 nM T44068 C6ULE4 44127480 EC50 = 190 nM T44068 C1LWJ0 44127481 EC50 = 710 nM T44068 CCI02W 44127575 EC50 = 550 nM T44068 CL10EZ 44127677 EC50 = 1700 nM T44068 C73XYH 44127678 EC50 = 350 nM T44068 CZ5FG8 44127679 EC50 = 3100 nM T44068 CB1W9S 44127681 EC50 = 760 nM T44068 CY39CN 44127782 EC50 = 600 nM T44068 C2AV1K 44190762 IC50 = 4070 nM T44068 CLR40G 44219629 EC50 = 180 nM T44068 CZ2BO8 44219630 EC50 = 280 nM T44068 CW7D8Q 44219641 EC50 = 62 nM T44068 CQ94HI 44267518 IC50 = 37500 nM T44068 C27AGX 44268214 IC50 = 15 nM T44068 C9D7RS 44268249 IC50 = 15 nM T44068 C5E2MI 44268254 IC50 = 1000 nM T44068 CNQ7X8 44268266 IC50 = 81 nM T44068 CLR0X8 44268268 EC50 = 300 nM T44068 C9TB2F 44268273 EC50 = 3 nM T44068 C6NY3M 44268274 IC50 = 1000 nM T44068 CGJT32 44268275 IC50 = 1000 nM T44068 CZ3W8B 44268277 IC50 = 100 nM T44068 CLS1U8 44268281 IC50 = 1000 nM T44068 C6R8SP 44268295 IC50 = 1000 nM T44068 C0UG8A 44268305 IC50 = 10 nM T44068 C2AJI5 44268308 IC50 = 140 nM T44068 CY6X8E 44268320 IC50 = 150 nM T44068 CCH34M 44268322 IC50 = 900 nM T44068 CAD4P0 44268324 EC50 = 450 nM T44068 CI91WY 44268327 EC50 = 1200 nM T44068 CMU89C 44268341 IC50 = 9000 nM T44068 CS87PI 44268349 IC50 = 60 nM T44068 CB7F6R 44268352 IC50 = 830 nM T44068 CPNS03 44268358 IC50 > 10000 nM T44068 C9JZ5T 44268365 IC50 = 6.7 nM T44068 CP2G7C 44268367 IC50 = 25 nM T44068 C1S3AB 44268464 IC50 = 190 nM T44068 C29IOC 44268470 IC50 = 530 nM T44068 CI64OC 44268478 IC50 = 220 nM T44068 CU84BM 44268479 IC50 = 240 nM T44068 CQY09P 44268482 IC50 = 1000 nM T44068 CRV1T3 44268495 IC50 = 150 nM T44068 CU21DW 44268496 IC50 = 150 nM T44068 CWG2Q7 44268498 IC50 = 510 nM T44068 C4D1OQ 44268509 IC50 = 880 nM T44068 C3YGB4 44268520 IC50 = 190 nM T44068 C5TZ8J 44268534 IC50 = 220 nM T44068 CS73JY 44268539 IC50 = 730 nM T44068 CN8P2B 44268556 IC50 = 250 nM T44068 CES3Y9 44268563 IC50 = 340 nM T44068 CY5J3N 44268568 IC50 = 300 nM T44068 CREN46 44268569 IC50 = 740 nM T44068 C0BR2A 44268570 IC50 = 800 nM T44068 C9H1IF 44268571 IC50 = 260 nM T44068 CBZ7N6 44268572 IC50 = 1000 nM T44068 C2LYD1 44268604 IC50 = 200 nM T44068 CD7UZ0 44268605 IC50 = 540 nM T44068 CF3VU1 44268632 IC50 = 350 nM T44068 C6S7VB 44276727 IC50 = 186 nM T44068 CW7A6K 44280795 IC50 = 8500 nM T44068 CR8D7Y 44280858 IC50 = 9000 nM T44068 C4JLV9 44280860 IC50 = 55000 nM T44068 C49FOW 44280903 IC50 = 550 nM T44068 CM6C4J 44280904 IC50 = 2100 nM T44068 CJ1B9Z 44280957 IC50 = 30000 nM T44068 CM9R8D 44281037 IC50 = 10000 nM T44068 CPO25L 44281073 IC50 = 56000 nM T44068 CI4NE5 44281074 IC50 = 25000 nM T44068 CG7A5O 44281097 IC50 = 3500 nM T44068 CS84VC 44281218 IC50 = 4500 nM T44068 CIPT87 44281219 IC50 = 4000 nM T44068 C1S3HD 44281255 IC50 = 2000 nM T44068 CZT1Q6 44281276 IC50 = 2000 nM T44068 COB42G 44281277 IC50 = 2000 nM T44068 C28KLB 44281344 IC50 = 2000 nM T44068 C65JLA 44281371 IC50 = 1000 nM T44068 CD78QG 44281372 IC50 = 2500 nM T44068 CBNZ27 44281384 IC50 = 2000 nM T44068 CG3D5J 44281395 IC50 = 8000 nM T44068 CBL4F1 44281396 IC50 = 715 nM T44068 CO9F8Q 44281400 IC50 = 3660 nM T44068 CT0XW9 44281407 IC50 = 7000 nM T44068 CK3Z4L 44281408 IC50 = 2600 nM T44068 C7P3WY 44281424 IC50 = 2430 nM T44068 CIO1V4 44281425 IC50 = 3000 nM T44068 CJU5O2 44281467 IC50 = 2000 nM T44068 CI1C5Q 44281468 IC50 = 2000 nM T44068 CTL1G7 44281469 IC50 = 5000 nM T44068 CEN7H9 44281470 IC50 = 65000 nM T44068 CC90RN 44281530 IC50 = 3000 nM T44068 CLXI95 44281531 IC50 = 16000 nM T44068 C0DG5M 44285225 IC50 = 2000 nM T44068 CNO3I4 44285226 IC50 = 6000 nM T44068 C7L5MN 44285529 IC50 = 200 nM T44068 CUF3O2 44285634 IC50 = 350 nM T44068 CTIA64 44285685 IC50 = 7000 nM T44068 C0JY4C 44285692 IC50 = 37000 nM T44068 CPQ16U 44286964 Ki > 100000 nM T44068 CKL84D 44286965 Ki = 1250 nM T44068 C2IJ9G 44286980 Ki = 140000 nM T44068 CPN74V 44286983 Ki = 590 nM T44068 CE5GK6 44287268 Ki = 139000 nM T44068 CD0E2S 44287321 Ki = 243000 nM T44068 CA72HF 44287337 Ki = 310 nM T44068 CV0J2F 44288393 Ki = 24 nM T44068 C53RQT 44298256 IC50 = 600 nM T44068 C5EXK1 44298281 IC50 = 3000 nM T44068 C82TAV 44298288 IC50 = 1400 nM T44068 C0ICR9 44298290 IC50 = 4000 nM T44068 COTF72 44298306 IC50 = 10000 nM T44068 CX4QG5 44298314 IC50 = 330 nM T44068 CIJ6H2 44298315 IC50 = 580 nM T44068 CDCP96 44298497 IC50 = 1000 nM T44068 CNK60M 44298515 IC50 = 1400 nM T44068 CZHU81 44298516 IC50 = 4000 nM T44068 CJ1X0Z 44298533 IC50 = 2600 nM T44068 CRD69E 44298695 IC50 = 1800 nM T44068 CP72DS 44298700 IC50 = 9000 nM T44068 CSKD26 44298718 IC50 = 10000 nM T44068 CBW06V 44298728 IC50 = 40000 nM T44068 CVN75C 44298731 IC50 = 1000 nM T44068 C67YCD 44298752 IC50 = 10000 nM T44068 CO9BE8 44298761 IC50 = 100000 nM T44068 CYGM23 44298767 IC50 = 10000 nM T44068 CD51GN 44298769 IC50 = 1500 nM T44068 CE01UQ 44298781 IC50 = 970 nM T44068 CUK01S 44298787 IC50 = 650 nM T44068 CFRN96 44298821 IC50 = 4200 nM T44068 C40OYU 44298822 IC50 = 4000 nM T44068 C19XHR 44298823 IC50 = 2500 nM T44068 CSW8G0 44298843 IC50 = 1800 nM T44068 CQID30 44298849 IC50 = 700 nM T44068 C8FL6R 44298850 IC50 = 3000 nM T44068 CHJR57 44298851 IC50 = 220 nM T44068 C2GBS7 44298852 IC50 = 900 nM T44068 C6GD9N 44301617 IC50 = 52000 nM T44068 CI0OY1 44301618 IC50 = 1500 nM T44068 C4P1OD 44301764 IC50 = 40000 nM T44068 CCH74I 44301803 IC50 = 3000 nM T44068 C3T9OF 44301804 IC50 = 6500 nM T44068 CY63AQ 44301805 IC50 = 7000 nM T44068 CA3VZ2 44301806 IC50 = 6000 nM T44068 C2OJ3N 44301818 IC50 = 1100 nM T44068 CNZ68T 44301819 IC50 = 1600 nM T44068 CMFW56 44301831 IC50 = 7000 nM T44068 CJB9L8 44301832 IC50 = 3700 nM T44068 C4DZ6V 44301842 IC50 = 13000 nM T44068 CW02XN 44301843 IC50 = 9000 nM T44068 C6P8UW 44301866 IC50 = 850 nM T44068 C8T7OB 44301867 IC50 = 960 nM T44068 CS4ET3 44301880 IC50 = 90000 nM T44068 CM4G9Z 44301881 IC50 = 100000 nM T44068 C6VDZ8 44301886 IC50 = 50000 nM T44068 C08SKL 44301979 IC50 = 19000 nM T44068 C8EGA1 44302005 IC50 = 30000 nM T44068 C9J6RY 44303192 IC50 = 10000 nM T44068 CN0DE9 44303198 IC50 = 1000 nM T44068 CA4BQ1 44306956 IC50 = 290 nM T44068 C70GLV 44306959 IC50 = 5300 nM T44068 C9HL3E 44306979 IC50 = 2000 nM T44068 C75OJI 44306985 IC50 = 2000 nM T44068 CH58SX 44306991 IC50 = 6300 nM T44068 C0XI5A 44306992 IC50 = 10000 nM T44068 CN23SP 44307007 IC50 = 1000 nM T44068 C4LRJ3 44307063 IC50 = 2000 nM T44068 CYI2V9 44307064 IC50 = 1000 nM T44068 C7KWF2 44307065 IC50 = 1000 nM T44068 C3H9QV 44307113 IC50 = 80 nM T44068 CC4IL0 44307144 IC50 = 600 nM T44068 CK0WG5 44307166 IC50 = 910 nM T44068 CLB56U 44307186 IC50 = 590 nM T44068 CYX08L 44307196 IC50 = 470 nM T44068 CNCV21 44307205 IC50 = 900 nM T44068 C5Q4MP 44307333 IC50 = 5500 nM T44068 CVK8S0 44307340 IC50 = 440 nM T44068 C1RYI9 44307343 IC50 = 1000 nM T44068 CK1P5Z 44307378 IC50 = 1300 nM T44068 CV1Z0F 44307379 IC50 = 1300 nM T44068 C5NIP7 44307396 IC50 = 860 nM T44068 C9G4UO 44309272 EC50 = 12 nM T44068 CKWA37 44309523 EC50 = 1600 nM T44068 CMJX34 44309649 EC50 = 10300 nM T44068 CFHD64 44312269 Ki = 6400 nM T44068 CVX04Z 44312421 Ki = 440 nM T44068 CF3H5U 44312924 EC50 = 6100 nM T44068 CY4K0A 44312949 IC50 = 1000 nM T44068 C3L4PJ 44313090 IC50 = 1000 nM T44068 CL2UV6 44313150 EC50 = 10000 nM T44068 CPA5B7 44313161 IC50 = 6500 nM T44068 C15EMW 44328703 EC50 = 316.23 nM T44068 CV8J4A 44331302 EC50 = 3160 nM T44068 C97IJY 44331346 EC50 = 730 nM T44068 C0RDZ3 44331351 EC50 = 520 nM T44068 CIFO93 44331425 EC50 = 1860 nM T44068 C5Y8GN 44331426 EC50 = 580 nM T44068 CU4EQ5 44331443 EC50 = 520 nM T44068 CWE69G 44331444 EC50 = 6300 nM T44068 CI17GW 44331766 EC50 = 417 nM T44068 CR36NA 44335496 IC50 = 7000 nM T44068 C5BX2N 44335497 IC50 = 20000 nM T44068 CD7ZV4 44335498 IC50 = 10000 nM T44068 C9UE7G 44335499 IC50 = 30000 nM T44068 CDS5L1 44335534 IC50 = 160 nM T44068 C7MC1U 44335548 IC50 = 970 nM T44068 CY7LH9 44335560 IC50 = 2000 nM T44068 C6IA8P 44335562 IC50 = 10000 nM T44068 CLE91U 44335572 IC50 = 10000 nM T44068 C4B8OE 44335588 IC50 = 60000 nM T44068 C17PHB 44335589 IC50 = 2000 nM T44068 C7A4UT 44335603 IC50 = 8000 nM T44068 CFX90I 44335618 IC50 = 2000 nM T44068 C14ILU 44335628 IC50 = 60000 nM T44068 CX8QZ4 44335651 IC50 = 30000 nM T44068 C03GDI 44335663 IC50 = 7000 nM T44068 CL2BX0 44335833 IC50 = 100000 nM T44068 C4M8EN 44335844 IC50 = 100000 nM T44068 C3DP9K 44335882 IC50 = 100000 nM T44068 CM0XE7 44336180 EC50 = 460 nM T44068 CNW2Y0 44336319 EC50 = 2640 nM T44068 C4PU1O 44349588 IC50 = 110 nM T44068 CS1L9V 44349629 IC50 = 740 nM T44068 CO27RQ 44349645 IC50 = 620 nM T44068 C6WP1E 44349646 IC50 = 74 nM T44068 CZK46C 44369602 EC50 < 10000 nM T44068 C3M7BC 44377315 IC50 = 1000 nM T44068 CS6C8L 44377316 IC50 = 4000 nM T44068 CI1MN9 44377412 IC50 = 10000 nM T44068 CEW6J9 44377513 IC50 = 2000 nM T44068 C8DYK5 44377514 IC50 = 850 nM T44068 CRB49F 44377517 IC50 = 10000 nM T44068 C3XLD1 44377636 IC50 = 5000 nM T44068 C3BQ1X 44377637 IC50 = 2000 nM T44068 CHB6Q2 44377650 IC50 = 10000 nM T44068 CNEO30 44377665 IC50 = 50000 nM T44068 CKI9O8 44377677 IC50 = 10000 nM T44068 CQEA58 44377687 IC50 = 3000 nM T44068 C49FSC 44377753 IC50 = 27000 nM T44068 CW42ZY 44377754 IC50 = 5300 nM T44068 C04XMY 44377755 IC50 = 100000 nM T44068 C02ZPF 44377957 IC50 = 10000 nM T44068 CG2F6I 44386630 Ki = 3.8 nM T44068 CQ3OE6 44392175 EC50 = 0.9 nM T44068 C0S9HV 44392181 EC50 = 12 nM T44068 C82SPF 44392190 EC50 = 3 nM T44068 CE2M3X 44392212 EC50 = 3.6 nM T44068 CDF75J 44392215 EC50 = 2.2 nM T44068 CO43RV 44392228 EC50 = 15 nM T44068 C96SHC 44392230 EC50 = 1.3 nM T44068 C37GEF 44392240 EC50 = 51 nM T44068 CYEF45 44392255 EC50 = 27 nM T44068 C0CBD4 44392457 EC50 = 10 nM T44068 CXO92R 44392490 EC50 = 120 nM T44068 C7QJN5 44392542 EC50 = 7.6 nM T44068 CND67K 44392552 EC50 = 13 nM T44068 CS3H7D 44392558 EC50 = 36 nM T44068 C83OKR 44392575 EC50 = 9.6 nM T44068 CI4J7L 44396488 EC50 = 19 nM T44068 CB37RE 44396513 EC50 = 6.2 nM T44068 C6HQL1 44396521 EC50 = 29 nM T44068 CE1MS4 44396530 EC50 = 7.3 nM T44068 C2YP6O 44396531 EC50 = 5.6 nM T44068 CLYG39 44396532 EC50 = 21 nM T44068 CN7HX8 44396568 EC50 = 19 nM T44068 C2DOA1 44396577 EC50 = 6.6 nM T44068 CHXA19 44396596 EC50 = 6.6 nM T44068 CZ71YN 44396659 Ki = 230 nM T44068 CW4OR6 44396715 EC50 = 1.3 nM T44068 C4BXY6 44396729 Ki = 89 nM T44068 CRY62C 44396736 EC50 = 1.2 nM T44068 C4WO2Y 44396737 EC50 = 58 nM T44068 C6CZX4 44396738 EC50 = 85 nM T44068 CUO7X8 44396779 EC50 = 3.1 nM T44068 C53GBI 44396798 EC50 = 26 nM T44068 C0EXA1 44407083 IC50 > 10000 nM T44068 CG87PW 44409290 Ki > 1000 nM T44068 CSA2X5 44419254 EC50 > 10000 nM T44068 CG5XU6 44419315 EC50 > 10000 nM T44068 C4ABS0 44419316 EC50 > 10000 nM T44068 CQ89AE 44419324 EC50 > 10000 nM T44068 CFG74O 44419332 EC50 = 8.7 nM T44068 C5YBA0 44423639 Ki > 100000 nM T44068 C3XR8N 44423640 Ki = 61.1 nM T44068 C45ISV 44423641 Ki = 6460 nM T44068 CK1XO7 44423643 Ki = 23.2 nM T44068 CD72TX 44423644 Ki = 1110 nM T44068 C34MXL 44423645 Ki = 66.7 nM T44068 C7IAO1 44423646 Ki = 2160 nM T44068 C5P4OW 44433250 Ki = 7.92 nM T44068 CKZF16 44439165 Ki = 2511.89 nM T44068 CA4HZ3 44439167 Ki = 1584.89 nM T44068 CN8G6D 44441226 EC50 = 12.59 nM T44068 C4Q1JB 44441227 EC50 = 158.49 nM T44068 CC34NU 44441228 EC50 = 19.95 nM T44068 CE34HD 44441229 EC50 = 79.43 nM T44068 CXE23W 44441230 EC50 = 12.02 nM T44068 CZ96SJ 44441231 EC50 = 100 nM T44068 CTWM30 44441232 EC50 = 25.12 nM T44068 CA8E5H 44441233 EC50 = 398.11 nM T44068 CP2H0M 44441234 EC50 = 19.95 nM T44068 CZ2K7C 44441235 EC50 = 100 nM T44068 CR9B1F 44441236 EC50 = 3981.07 nM T44068 C6MFP8 44444153 EC50 > 10000 nM T44068 C1QZW9 44444154 EC50 > 10000 nM T44068 CGDZ68 44444166 EC50 > 10000 nM T44068 C9OIT6 44444167 EC50 > 10000 nM T44068 CG2QI4 44444169 EC50 > 10000 nM T44068 C58UHL 44444170 Ki > 10000 nM T44068 CUAN40 44444171 EC50 > 10000 nM T44068 CVQ59T 44444172 EC50 > 10000 nM T44068 C60YDC 44444173 EC50 = 58.3 nM T44068 C1IB7H 44444175 EC50 > 10000 nM T44068 CZ0VJ5 44444176 EC50 > 10000 nM T44068 CD74SN 44444179 Ki = 1500 nM T44068 C5TM3W 44444185 Ki = 1000 nM T44068 C16XQT 44444187 Ki = 730 nM T44068 C6PS3A 44444188 Ki = 570 nM T44068 CZAK23 44444189 Ki = 490 nM T44068 C9A3KP 44444191 Ki = 270 nM T44068 CA08VR 44444193 Ki = 420 nM T44068 CNS8K2 44444195 Ki = 1050 nM T44068 C0SA8C 44444378 Ki = 120 nM T44068 C9QP8S 44444393 Ki = 1550 nM T44068 C12XGE 44456400 Ki > 10000 nM T44068 C1A6ZC 44457929 EC50 = 370 nM T44068 C7O0IE 44458134 IC50 = 5000 nM T44068 C68NOT 44461468 IC50 = 10000 nM T44068 CDZ56W 44461485 IC50 > 10000 nM T44068 CM5ZH4 44461486 IC50 = 8500 nM T44068 C2GZ3R 44461488 IC50 = 100000 nM T44068 C1L6GN 44461489 IC50 = 10000 nM T44068 CQ8UE4 44461716 IC50 = 2000 nM T44068 C4TMP7 44461717 IC50 = 2000 nM T44068 C39FRG 44461718 IC50 = 5500 nM T44068 CM4F7J 44461719 IC50 = 10000 nM T44068 C4DL5C 44469677 IC50 > 10000 nM T44068 C2QK4J 44472590 IC50 > 20000 nM T44068 CQ8C3F 44472591 IC50 > 20000 nM T44068 CC2TA5 44472592 IC50 > 20000 nM T44068 CWN95E 44472610 IC50 > 20000 nM T44068 C1H2ZT 44472612 IC50 > 20000 nM T44068 C9G5ID 44472613 IC50 > 20000 nM T44068 C5N4KE 44472633 IC50 > 20000 nM T44068 CEH82X 44472636 IC50 > 20000 nM T44068 CMH3J4 44472637 IC50 > 20000 nM T44068 CC6G0Z 44517692 EC50 = 90 nM T44068 C5BYX7 44517694 EC50 = 70 nM T44068 CY8PO3 44517696 EC50 = 70 nM T44068 CS8G3O 44560739 EC50 > 1000 nM T44068 CE18ZY 44560791 EC50 = 75 nM T44068 C7V8EF 44560792 EC50 = 80 nM T44068 CMP8T6 44560793 EC50 = 190 nM T44068 CP36SU 44560794 EC50 = 24 nM T44068 C9P7BS 44565907 EC50 = 93 nM T44068 CP0JB5 44565908 EC50 = 200 nM T44068 CAF8L7 44565931 EC50 = 140 nM T44068 CDUZ13 44565932 EC50 = 390 nM T44068 CBD52U 44574651 EC50 = 1300 nM T44068 CSGI84 44574685 EC50 > 100000 nM T44068 CIF02K 44574686 EC50 = 120000 nM T44068 C4PN5S 44574687 EC50 = 180 nM T44068 C6BVQ7 44574688 EC50 = 280 nM T44068 C6UTI8 44574720 EC50 = 250 nM T44068 C0RB7H 44574721 EC50 = 330 nM T44068 C56UZO 44574722 EC50 = 280 nM T44068 CVP31K 44574723 EC50 = 43 nM T44068 CM53PL 44574757 EC50 = 2500 nM T44068 CLG2N1 44574758 EC50 = 9600 nM T44068 C6E2SN 44574759 EC50 = 650 nM T44068 CIS5B4 44574825 EC50 = 140 nM T44068 CK2H8G 44574826 EC50 = 130 nM T44068 CU7H5I 44574827 EC50 = 270 nM T44068 C9GZ3R 44574867 EC50 = 190 nM T44068 CL7SJ3 44574868 EC50 = 260 nM T44068 C9HE8U 44574913 EC50 = 500 nM T44068 CO3V6F 44574978 EC50 = 170 nM T44068 CKE82M 44579649 EC50 = 690 nM T44068 C0OHE7 44579650 EC50 = 190 nM T44068 CS92ZG 44579651 EC50 = 28 nM T44068 CA5O2G 44579925 EC50 = 64 nM T44068 C90FXY 44579940 EC50 = 240 nM T44068 CUZ85X 44579941 EC50 > 1000 nM T44068 CLU26M 44579964 EC50 > 100 nM T44068 C81ALE 44579965 EC50 > 100 nM T44068 C6LV4K 44579966 EC50 = 140 nM T44068 CZL47Y 44580009 EC50 = 550 nM T44068 C86TQI 44580010 EC50 = 510 nM T44068 C8C0FP 44580011 EC50 = 380 nM T44068 CTE0P6 44580039 EC50 = 130 nM T44068 CZ3OG8 44580040 EC50 = 620 nM T44068 C5YB0H 44580041 EC50 = 190 nM T44068 CBH97I 44580042 EC50 = 840 nM T44068 C3L5ER 44583033 EC50 = 3 nM T44068 CXD63G 44589133 EC50 = 2035 nM T44068 CS08ED 44589400 EC50 = 7282 nM T44068 CJ0D9X 44591506 EC50 = 130 nM T44068 C32HSU 44591507 EC50 = 150 nM T44068 CWQ2K4 44591508 EC50 = 39 nM T44068 CC18SZ 45101519 EC50 = 1.8 nM T44068 CL9UT7 45101520 EC50 = 4.5 nM T44068 C04EWA 45101521 EC50 = 24 nM T44068 CWIL37 45101522 EC50 = 9.9 nM T44068 C7CM3S 45101537 EC50 = 290 nM T44068 C07LMT 45267257 EC50 = 30 nM T44068 C7OTL6 45267631 EC50 > 1000 nM T44068 C5P2KR 45268128 EC50 = 50 nM T44068 C7NC2T 45268136 EC50 = 80 nM T44068 C9SIW5 45268516 EC50 = 150 nM T44068 C7GPS1 45269025 EC50 = 30 nM T44068 C2D7EA 45269373 EC50 > 1000 nM T44068 CEA21T 45269853 EC50 = 110 nM T44068 C5EO1Y 45270197 EC50 > 1000 nM T44068 CH2Y3X 45270673 EC50 = 40 nM T44068 CW2FT8 45270680 EC50 = 110 nM T44068 C43UZN 45270690 EC50 = 60 nM T44068 CCZ10H 45270697 EC50 = 130 nM T44068 CGTY98 45271036 EC50 = 130 nM T44068 CG2L0D 45271492 EC50 = 20 nM T44068 CK48MV 45271517 EC50 = 70 nM T44068 C13VYN 45271518 EC50 = 60 nM T44068 CMU01B 45271523 EC50 = 100 nM T44068 C0QOW1 45271886 EC50 = 73 nM T44068 CS27QE 45272430 EC50 = 90 nM T44068 CL76SG 45272431 EC50 = 70 nM T44068 C07GYE 45272758 EC50 > 1000 nM T44068 CBKW49 45273268 EC50 = 10 nM T44068 C6GW4V 45273276 EC50 = 56 nM T44068 CH10SC 45273280 EC50 = 40 nM T44068 CPJB52 45280075 EC50 > 10000 nM T44068 CZEB18 45375919 EC50 = 253 nM T44068 C6QES8 45380471 EC50 > 10000 nM T44068 CZ73IE 45381852 EC50 > 10000 nM T44068 CNI72R 45381932 EC50 > 10000 nM T44068 C0CHF4 45482789 IC50 = 5760 nM T44068 C7RYF5 45483810 EC50 = 0.8 nM T44068 C70MIX 45483813 EC50 = 0.6 nM T44068 C6IU9K 45483814 EC50 = 3.6 nM T44068 CJ5LO8 45483815 EC50 = 33 nM T44068 C1W0IA 45483816 EC50 = 5 nM T44068 CKY85H 45483825 EC50 > 10000 nM T44068 CVI32P 45483830 EC50 = 294 nM T44068 CI96VQ 45483831 EC50 > 10000 nM T44068 CNX06B 45483838 EC50 = 1869 nM T44068 CBN09R 45483839 EC50 = 695 nM T44068 CC3F7O 45483843 EC50 = 5.6 nM T44068 CH1BC2 45483844 EC50 = 6.7 nM T44068 CAZ4C7 45483846 EC50 = 26.5 nM T44068 CEH1G2 45483847 EC50 = 5 nM T44068 C4ISE8 45483848 EC50 = 1004 nM T44068 CGD86T 45483849 EC50 = 645 nM T44068 CSQT68 45483852 EC50 = 7.2 nM T44068 CN1KI6 45483864 EC50 = 3.7 nM T44068 C43ETK 45483868 EC50 = 3.7 nM T44068 C9QR8M 45484536 EC50 = 4.6 nM T44068 CN2L9F 45484537 EC50 = 28 nM T44068 C4JH6P 45484558 EC50 = 18 nM T44068 CS5RA6 45484568 EC50 = 5.3 nM T44068 C8YBJ6 45484569 EC50 = 5.7 nM T44068 CHQ83C 45484583 EC50 = 3.4 nM T44068 CQ07ZN 45484584 EC50 = 3.5 nM T44068 CI0M5N 45484646 EC50 = 11 nM T44068 C4U3XI 46232768 EC50 = 35 nM T44068 CI35QZ 46232769 EC50 = 4.5 nM T44068 C1TS7M 46232815 EC50 = 989.5 nM T44068 CE79ZN 46232816 EC50 = 207 nM T44068 CAF43W 46232856 EC50 = 436.5 nM T44068 CW1M4Q 46232857 EC50 = 240 nM T44068 CO2B9C 46232973 EC50 = 27 nM T44068 CF1B6A 46232974 EC50 = 2725 nM T44068 CSNR69 46233013 EC50 = 278.4 nM T44068 C7NA1H 46832227 EC50 > 25118.86 nM T44068 CNA42V 46832232 EC50 = 12.59 nM T44068 CN7MG5 46832505 EC50 = 31.62 nM T44068 CJ5B4A 46832507 EC50 = 19.95 nM T44068 CW0JV6 46832509 EC50 = 12.59 nM T44068 C7TN0H 46832510 EC50 = 398.11 nM T44068 C04XPW 46832798 EC50 = 12.59 nM T44068 CQ1BJ4 46832804 EC50 = 100 nM T44068 C6VS1A 46833102 EC50 = 50.12 nM T44068 CSYQ43 46833103 EC50 = 79.43 nM T44068 CQ3TM8 46845697 IC50 > 20000 nM T44068 CJV15G 46845698 IC50 = 12000 nM T44068 C0DB5H 46845699 IC50 = 19000 nM T44068 C2D6ZI 46881527 IC50 > 20000 nM T44068 CIP0H2 46881528 IC50 > 20000 nM T44068 CZ0PU9 46881529 IC50 = 3000 nM T44068 CTV6U8 46881530 IC50 > 10000 nM T44068 CFA38Z 46881531 IC50 = 9600 nM T44068 CIJU02 46881573 IC50 = 19000 nM T44068 C4YNT0 46881574 IC50 = 3100 nM T44068 CV5R2L 46881575 IC50 = 7600 nM T44068 CULH08 46881576 IC50 = 600 nM T44068 CYLF92 46881614 IC50 > 20000 nM T44068 CT56SD 46881615 IC50 > 20000 nM T44068 CLB86Z 46881616 IC50 > 10000 nM T44068 CJ1VO4 46881617 IC50 = 8300 nM T44068 C6D5IZ 46881618 IC50 = 1500 nM T44068 CTC02J 46881650 IC50 > 10000 nM T44068 CN9TK8 46881651 IC50 = 1100 nM T44068 CWZ4H5 46881652 IC50 > 10000 nM T44068 CZQ6C8 46881653 IC50 > 20000 nM T44068 CD27OS 46881698 IC50 = 1400 nM T44068 CGP45C 46881699 IC50 = 3400 nM T44068 C7BPN3 46881700 IC50 = 3000 nM T44068 CMR6C9 46881701 IC50 = 3600 nM T44068 C8QS6V 46881750 IC50 = 8600 nM T44068 C8XST7 46881751 IC50 > 20000 nM T44068 CW60AO 46881752 IC50 = 840 nM T44068 CFIE98 46881753 IC50 = 11000 nM T44068 C4EOF8 46881796 IC50 = 16000 nM T44068 C9HO2J 46881797 IC50 > 20000 nM T44068 CX8ZS6 46881798 IC50 > 20000 nM T44068 C9OE3N 46881799 IC50 > 20000 nM T44068 CV75XD 46881838 IC50 > 20000 nM T44068 CVR9M2 46881839 IC50 > 20000 nM T44068 C4D1XF 46881840 IC50 > 20000 nM T44068 CK0N6A 46881869 IC50 > 20000 nM T44068 C9CUP4 46881870 IC50 > 20000 nM T44068 C53CIB 46881871 IC50 > 20000 nM T44068 CGZ7K5 46881872 IC50 = 700 nM T44068 CHJ9D1 46881899 IC50 = 13000 nM T44068 C4D7PW 46881900 IC50 = 4900 nM T44068 CI7Q6U 46881901 IC50 = 1900 nM T44068 CTX8N0 46881902 IC50 > 20000 nM T44068 CR1H5N 46881935 IC50 > 10000 nM T44068 CQ87KZ 46881936 IC50 > 10000 nM T44068 CKDO83 46881937 IC50 = 5000 nM T44068 C7W1LE 46881938 IC50 = 6000 nM T44068 CXDJ80 46881980 IC50 > 10000 nM T44068 CP5O9V 46881981 IC50 = 12000 nM T44068 C4N0KV 46881982 IC50 = 2400 nM T44068 C50CFL 46881983 IC50 = 1700 nM T44068 C50GNW 46882028 IC50 = 9800 nM T44068 CBC6Z5 46882029 IC50 > 10000 nM T44068 C2Y3DO 46882030 IC50 = 4100 nM T44068 CWG7Z8 46882031 IC50 = 4000 nM T44068 CWI86A 46882084 IC50 = 1900 nM T44068 CBN3V6 46889642 Ki = 4530 nM T44068 CG72PB 46889643 Ki = 27 nM T44068 C8S4LM 46889670 Ki = 7 nM T44068 CEF90S 46889699 Ki = 1050 nM T44068 CH4Z0F 46889700 Ki = 240 nM T44068 C8K6HX 46889701 Ki = 170 nM T44068 CAO57K 46889727 Ki = 300 nM T44068 CTP3E7 46889728 Ki = 209 nM T44068 CW9LS6 46889729 Ki = 190 nM T44068 C7RI4K 46889730 Ki = 720 nM T44068 C4ISX8 46889767 Ki = 440 nM T44068 C3ZY5J 46889768 Ki = 245 nM T44068 C3F4IQ 46889769 Ki = 260 nM T44068 C1P5WV 46889770 Ki = 89 nM T44068 C02HNI 46889771 EC50 = 80 nM T44068 C4D5FH 46889772 Ki = 0.1 nM T44068 CKIM07 46889809 Ki = 76 nM T44068 C6CY1S 46889810 Ki = 14 nM T44068 C26WTA 46889811 Ki = 3.4 nM T44068 C2GC4K 46889812 Ki = 1 nM T44068 C9P4TD 46889852 Ki = 16 nM T44068 C1YVO4 46889853 Ki = 13 nM T44068 CFY40T 46889854 Ki = 32 nM T44068 CK8V2H 49800025 EC50 = 39.81 nM T44068 CV5G1H 49861320 EC50 = 250 nM T44068 C6OQV2 49862237 Ki > 1000 nM T44068 CX5TY8 49864332 Ki = 169 nM T44068 C3GAQ5 49864333 Ki = 1.5 nM T44068 CN9R1Z 49864334 Ki = 39.3 nM T44068 CP6XL8 49864335 Ki = 9.2 nM T44068 CCO9X4 49864355 Ki = 35.4 nM T44068 CO4BD7 49864356 Ki = 3.8 nM T44068 C5KHJ2 49864357 Ki = 902 nM T44068 C9NOK6 49864358 Ki = 2 nM T44068 CY0FL3 49864377 Ki = 112 nM T44068 CN87YW 49864378 Ki = 58.2 nM T44068 CEQI63 49864379 Ki = 15 nM T44068 CJ04XU 49864380 Ki = 1.4 nM T44068 CD48CK 49864381 Ki = 33.7 nM T44068 C7MZC6 49864394 Ki = 78.8 nM T44068 C7C8PK 49864395 Ki = 0.9 nM T44068 C5O7HP 49864396 Ki = 17 nM T44068 CLK3Y5 49864397 Ki = 6.9 nM T44068 C87HDG 49864412 Ki = 40.4 nM T44068 C8KVZ6 49864413 Ki = 1059 nM T44068 CUR2Z4 49864414 Ki = 1511 nM T44068 CVA6H4 49864415 Ki = 450 nM T44068 C8U7ID 49864416 Ki = 123 nM T44068 CFA63G 49864439 Ki = 662 nM T44068 CQVR67 49864440 Ki = 187 nM T44068 CZV9N8 49864441 Ki = 17.8 nM T44068 C62FLG 49864442 Ki = 8.4 nM T44068 CJQI64 49864443 Ki > 1000 nM T44068 C6SL3T 49864460 Ki = 1.7 nM T44068 C1WL8J 49864461 Ki = 31.3 nM T44068 C2RY0J 50878551 Ki > 10000 nM T44068 C1W6TV 50898777 Ki > 10000 nM T44068 CXMZ73 50898778 Ki > 10000 nM T44068 CLY9W1 50994950 IC50 > 20000 nM T44068 C2CH1R 50995330 IC50 > 20000 nM T44068 CE4KP1 51050257 Ki > 10000 nM T44068 CYR21W 51346867 IC50 = 2189 nM T44068 C4Z2FY 51347436 IC50 > 20000 nM T44068 CQG7X2 51349173 EC50 > 10000 nM T44068 C1F0DX 52941476 Ki = 289 nM T44068 CZMS46 52941603 Ki = 2902 nM T44068 C83BMV 52943362 Ki = 33 nM T44068 C3B2OF 52943383 Ki = 996 nM T44068 C61ZLX 52943770 Ki = 8560 nM T44068 CE13YX 52943919 Ki = 150 nM T44068 C5TW1N 52943932 Ki = 700 nM T44068 CVE5Q9 52943968 EC50 = 110 nM T44068 C69LKY 52943969 Ki = 2018 nM T44068 CP6U9S 52944986 Ki = 433 nM T44068 C0TWA8 52946357 Ki = 4980 nM T44068 CFX1D5 52946430 Ki = 1427 nM T44068 CI2PT6 52946537 Ki = 30 nM T44068 C7ULQ8 52947060 Ki = 230 nM T44068 CHK30N 52947443 Ki = 293 nM T44068 CD7EW1 52947562 EC50 = 5 nM T44068 CED37H 52948056 EC50 = 6.6 nM T44068 C04PTF 52948728 Ki = 4880 nM T44068 C6E9TK 52948792 Ki = 462 nM T44068 CU1R7B 52948805 Ki = 100 nM T44068 CI7S6O 52949488 EC50 = 9.6 nM T44068 CMX86D 52949489 EC50 = 450 nM T44068 C9VYT6 52949934 Ki = 450 nM T44068 C57DOH 53318280 IC50 = 1040 nM T44068 CJAH78 53319639 IC50 = 1520 nM T44068 CA45EM 53326195 IC50 = 2930 nM T44068 C9SDC2 53326196 IC50 = 1780 nM T44068 CM5WF2 53326197 IC50 = 242 nM T44068 C3EAT2 53326839 IC50 = 2150 nM T44068 CLN6B9 53357711 EC50 = 125.89 nM T44068 CL7US4 53357712 EC50 = 199.53 nM T44068 C7WKR1 53387673 Ki = 3000 nM T44068 CFB1N5 53387674 Ki = 2300 nM T44068 C9DGX4 53494950 IC50 = 0.04 nM T44068 CWYX94 54757772 EC50 > 10000 nM T44068 CRGV73 56597179 EC50 = 3.631 nM T44068 CB8O9W 56598831 EC50 = 9.772 nM T44068 CQKF90 56598832 EC50 = 2.291 nM T44068 CR6PU5 56598833 EC50 = 22.91 nM T44068 CRO1Y2 56598967 EC50 = 4.467 nM T44068 C43AZK 56658246 EC50 = 251.19 nM T44068 CCAE43 56658405 EC50 = 31.62 nM T44068 CMWZ90 56658407 EC50 = 7.943 nM T44068 CU2C6F 56663238 EC50 = 39.81 nM T44068 CPE84D 56665368 EC50 = 31.62 nM T44068 CEU7B9 56668796 EC50 = 10 nM T44068 C0CS2Z 56670092 EC50 = 199.53 nM T44068 C7D6LT 56670158 EC50 = 39.81 nM T44068 C9CRA4 56672269 EC50 = 31.62 nM T44068 CM3YO8 56672271 EC50 = 31.62 nM T44068 CXC4G1 56673609 EC50 = 158.49 nM T44068 CRSF93 56673674 IC50 = 794.33 nM T44068 CLB1V0 56675663 EC50 = 50.12 nM T44068 CE5DQ6 56678849 EC50 = 50.12 nM T44068 CT2E1Z 56678973 EC50 = 7.943 nM T44068 C6T7YR 56943485 EC50 = 12.59 nM T44068 C7DEO8 56943515 EC50 = 6.31 nM T44068 CZF4B5 56943517 EC50 = 7.943 nM T44068 CJ81YS 56943518 EC50 = 7.943 nM T44068 C5M0CT 56943545 EC50 = 7.943 nM T44068 CMUQ15 56943546 EC50 = 7.943 nM T44068 C1TC7Q 56963799 Ki > 10000 nM T44068 C53OMP 57391554 IC50 = 63.1 nM T44068 CYZD14 57395043 IC50 > 3162.28 nM T44068 C2CEB9 57398562 IC50 = 501.19 nM T44068 C1NGZ7 57400229 IC50 = 199.53 nM T44068 C3TYE1 57401435 IC50 = 3162.28 nM T44068 CM7EN2 57401436 IC50 = 1258.93 nM T44068 CNYB81 59119410 Ki = 15848.93 nM T44068 CW09LS 59119417 Ki = 12589.25 nM T44068 CB47FI 59119455 Ki = 12589.25 nM T44068 CI3VH0 59119466 Ki = 10000 nM T44068 CI9P1B 59119467 Ki = 12589.25 nM T44068 C4UF6I 59119472 Ki = 25118.86 nM T44068 C3WS7G 59707188 EC50 > 10000 nM T44068 CGO41Y 59707195 EC50 > 10000 nM T44068 C5BSH0 66653268 EC50 = 3.02 nM T44068 CS2K0M 66796015 EC50 = 7.943 nM T44068 C3ARI1 67972106 IC50 > 20000 nM T44068 CXJ68U 67972107 IC50 > 20000 nM T44068 CB05ID 67972431 IC50 > 20000 nM T44068 CMG51Y 68807656 Ki = 5.5 nM T44068 CPX1H7 69119729 EC50 = 501.19 nM T44068 CV57BY 69119831 EC50 = 158.49 nM T44068 C86CXO 69119890 EC50 = 251.19 nM T44068 C4H3LN 69120058 EC50 = 1000 nM T44068 CNVH59 69442961 EC50 = 1995.26 nM T44068 CKWP40 69447283 EC50 = 1995.26 nM T44068 CAQ94I 70680981 IC50 = 1.5 nM T44068 C5Z4DK 70680982 IC50 = 0.3 nM T44068 CB9IM4 70680983 IC50 = 20 nM T44068 C49TOI 70680984 IC50 = 0.14 nM T44068 C5XHF2 70683106 IC50 = 0.25 nM T44068 CDEU50 70683107 IC50 = 2 nM T44068 CYC6X2 70683108 IC50 = 0.1 nM T44068 CH6KU0 70683109 IC50 = 0.05 nM T44068 CONA38 70684846 Ki = 183 nM T44068 C3I6XB 70685188 IC50 = 10 nM T44068 CDCJ06 70687345 IC50 = 0.2 nM T44068 CA56KM 70687346 IC50 > 100 nM T44068 C1OMH5 70687347 IC50 = 10 nM T44068 CR40KF 70687348 IC50 = 5 nM T44068 C7LTF2 70689402 IC50 = 1 nM T44068 C02NQY 70691181 Ki = 259 nM T44068 C7FY3A 70691507 IC50 = 0.1 nM T44068 C9XB6R 70691508 IC50 = 26 nM T44068 CJ6CU7 70693598 IC50 = 21 nM T44068 CFZI26 70693599 IC50 = 2 nM T44068 CRP9N3 70693600 IC50 = 0.05 nM T44068 CIS85K 70693601 IC50 = 0.35 nM T44068 CSL0X3 70695718 IC50 = 3 nM T44068 CBDL19 70792359 IC50 > 20000 nM T44068 CI0GU8 71660496 IC50 > 48500 nM T44068 CWH6T3 72548703 IC50 = 297 nM T44068 CC65OA 73213195 Ki > 10000 nM T44068 CW83DK 73213196 Ki > 10000 nM T44068 C7TM8S 73349644 EC50 = 100 nM T44068 C74QNU 73352659 EC50 = 60 nM T44068 CG0Z2D 73357212 EC50 = 30 nM T44068 C2E7QW 75201901 Ki = 7600 nM T44068 CVY13Q 76314766 IC50 > 20000 nM T44068 C5ZDK4 76315637 EC50 = 7.2 nM T44068 CFZU52 76315638 EC50 = 19 nM T44068 C0X7CQ 76315639 EC50 = 69 nM T44068 CGZ5C4 76315640 EC50 = 22 nM T44068 C67YUD 76318362 IC50 > 20000 nM T44068 C1M4TQ 76318363 IC50 > 20000 nM T44068 CCUG71 76318364 IC50 > 20000 nM T44068 C9PM0U 76319327 EC50 = 6.8 nM T44068 CR05PL 76322043 IC50 > 20000 nM T44068 CQ3CW1 76322044 IC50 > 20000 nM T44068 CFU26T 76322045 IC50 = 4329 nM T44068 CTD25H 76322046 IC50 > 20000 nM T44068 C61AMT 76322047 IC50 > 20000 nM T44068 CI8XA7 76322965 EC50 = 44 nM T44068 CQI0H5 76325667 IC50 > 20000 nM T44068 C6R4BP 76325668 IC50 > 20000 nM T44068 CB71EI 76325669 IC50 > 20000 nM T44068 C03YTR 76329059 EC50 = 6309.57 nM T44068 CRW8C5 76329232 IC50 > 20000 nM T44068 C5SKR4 76332892 IC50 = 13340 nM T44068 CMR86G 76332893 IC50 > 20000 nM T44068 CTVI40 76332894 IC50 > 20000 nM T44068 CL7TN0 76332895 IC50 > 20000 nM T44068 C8PGV1 76333795 EC50 = 13 nM T44068 CQ47BW 76336499 IC50 > 20000 nM T44068 C92WBQ 76336500 IC50 > 20000 nM T44068 C8KBZ1 76336501 IC50 > 20000 nM T44068 CQM69X 76336502 IC50 > 20000 nM T44068 CZM89H 90644139 Ki = 7943.28 nM T44068 C0N3TA 90644140 Ki = 39810.72 nM T44068 CP14DT 90644141 Ki = 7943.28 nM T44068 C93QFA 90644142 Ki > 10000 nM T44068 CE48KB 90644143 Ki > 10000 nM T44068 CW95JO 90644144 Ki > 10000 nM T44068 C3T1UD 90644145 Ki > 10000 nM T44068 CN8SF5 90644146 Ki = 79432.82 nM T44068 CB7I0W 90644147 Ki = 125892.54 nM T44068 CZ60EK 90644148 Ki = 125892.54 nM T44068 CEZ23R 90644149 Ki > 10000 nM T44068 C9DTM6 90644150 Ki > 10000 nM T44068 C4T1VR 90644151 Ki > 10000 nM T44068 C37DWQ 90644152 Ki > 10000 nM T44068 C57JOK 90644153 Ki = 6309.57 nM T44068 C6C2HF 90644154 Ki = 31622.78 nM T44068 CNXH73 90645344 EC50 = 2.512 nM T44068 C9W1FB 90645345 EC50 = 12.59 nM T44068 CR7OT8 90645346 EC50 = 1.995 nM T44068 C9A5KY 90645347 EC50 = 1.585 nM T44068 C5UF4C 90666101 EC50 > 10000 nM T44068 CDI39M 90666102 EC50 > 10000 nM T44068 CU2FI1 90666103 EC50 > 10000 nM T44068 C18GXP 90666104 EC50 > 10000 nM T44068 C87KZI 90666105 EC50 > 10000 nM T44068 CBR34H 90666106 EC50 > 10000 nM T44068 CWG37L 90666107 EC50 > 10000 nM T44068 C30FIA 90666108 EC50 > 10000 nM T44068 CV61GN 90666109 EC50 > 10000 nM T44068 C0SIZ8 90666110 EC50 > 10000 nM T44068 C0FH6V 90666111 EC50 > 10000 nM T44068 CZ8I0G 90666112 EC50 > 10000 nM T44068 C6LB4R 90666113 EC50 > 10000 nM T44068 C5MCU0 90666114 EC50 > 10000 nM T44068 C0ZCW5 90666115 EC50 > 10000 nM T44068 CC5I0L 90666116 EC50 > 10000 nM T44068 CIZ46C 90666117 EC50 > 10000 nM T44068 C7WR2F 90666118 EC50 > 10000 nM T44068 C6KU1V 90666119 EC50 > 10000 nM T44068 CK68NB 90666120 EC50 > 10000 nM T44068 CEV61D 90666121 EC50 > 10000 nM T44068 CZ4P0B 90666122 EC50 > 10000 nM T44068 CV52KY 90666123 EC50 > 10000 nM T44068 CZSB43 118710935 Ki = 6.9 nM T44068 CX6NP5 118710936 Ki = 18 nM T44068 CB5VH9 118710937 Ki = 40 nM T44068 CDJZ51 118710938 Ki = 391 nM T44068 CQ5Z8V 118710939 Ki = 62 nM T44068 CWGD39 118710940 Ki = 0.8 nM T44068 CL8SA7 118710941 Ki = 30 nM T44068 CEY68Q 118710942 Ki = 58 nM T44068 CM8P2H 118710943 Ki = 77 nM T44068 CHL2U8 118710944 Ki = 343 nM T44068 CVHK79 118710945 Ki = 33 nM T44068 CU68XQ 118710946 Ki = 438 nM T44068 CG8PJ0 118710947 Ki = 6.1 nM T44068 C3GW0U 118710948 Ki = 7.9 nM T44068 C9QB7F 118710949 Ki = 13 nM T44068 CMJ0S5 118710950 Ki = 4.3 nM T44068 C6I2UZ 118710951 Ki = 21 nM T44068 CQNL51 118725301 EC50 = 0.8128 nM T44068 C4D9QY 127026491 IC50 > 20000 nM T44068 CZ61LK 127034966 IC50 = 630.96 nM T44068 CA0SN5 127034967 IC50 = 199.53 nM T44068 CQ0ZT9 127035062 Ki = 1885 nM T44068 C7L1DB 127037832 IC50 > 20000 nM T44068 CG84RM 127041558 IC50 > 20000 nM T44068 CS20QX 127041559 IC50 > 20000 nM T44068 CN2T3I 127041869 IC50 > 20000 nM T44068 C2BE3M 127041870 IC50 > 20000 nM T44068 C31SDE 127042181 IC50 > 20000 nM T44068 CJ8GS7 127045855 EC50 = 39.81 nM T44068 C4D6BQ 127046950 EC50 = 501.19 nM T44068 C50GOC 130442480 Ki = 9600 nM T44068 CM04RF 130442572 Ki = 8500 nM T44068 CS58HX 132060734 Ki = 1894 nM T44068 C1GY2T 135156251 EC50 > 10000 nM T44068 C2QCA5 137631487 IC50 > 20000 nM T44068 C8HPN4 137634334 IC50 > 20000 nM T44068 CZ4TA9 137640201 Ki = 10232.93 nM T44068 C70XZQ 137643636 IC50 > 20000 nM T44068 CL06NY 137648464 IC50 > 20000 nM T44068 CUFO39 137649223 IC50 > 20000 nM T44068 C65XKJ 137653127 IC50 > 20000 nM T44068 C3LG7W 137655838 IC50 > 20000 nM T44068 CN2UE9 137656598 IC50 > 20000 nM T44068 C9C8LN 141465526 EC50 > 10000 nM T44068 CP6AM5 145949377 Ki > 100000 nM T44068 CROP78 145949554 Ki > 100000 nM T44068 C8XAH1 145950880 Ki > 100000 nM T44068 C53EGH 145950894 Ki > 100000 nM T44068 C87JIM 145951255 Ki = 10471.29 nM T44068 CQC79A 145951865 Ki > 100000 nM T44068 CUJ2G6 145952345 Ki > 100000 nM T44068 C0UBV8 145955012 Ki > 100000 nM T44068 CMGN62 145956070 Ki = 6606.93 nM T44068 CS93JU 145956073 Ki = 79432.82 nM T44068 CHXP91 145956144 Ki > 100000 nM T44068 CZK0L8 145956164 Ki > 100000 nM T44068 CRUI17 145956819 Ki = 15488.17 nM T44068 C6I1XE 145956976 Ki = 13489.63 nM T44068 CQO8H5 145958250 Ki > 100000 nM T44068 CC32ZJ 145958632 Ki > 100000 nM T44068 C29YFS 145959974 Ki = 26915.35 nM T44068 C9MSK2 145960116 Ki > 100000 nM T44068 C72IAC 145980824 EC50 > 10000 nM T44068 C8EHD9 145981007 EC50 > 10000 nM T44068 C4U3RO 145981079 EC50 = 1584.89 nM T44068 CU2LP6 145981405 EC50 > 10000 nM T44068 CBNQ70 145982607 EC50 = 36.81 nM T44068 C6MWR1 145982668 EC50 = 123.7 nM T44068 CFBS76 145983266 EC50 = 223.6 nM T44068 CZ60KX 145983355 EC50 = 298.8 nM T44068 COZ4J2 145983711 EC50 = 12700 nM T44068 C9DX1E 145984042 EC50 = 6204 nM T44068 CT4BM0 145984324 EC50 = 426.2 nM T44068 CE5PC2 145984584 EC50 = 2.884 nM T44068 C82AHK 145984792 EC50 = 100000 nM T44068 CH7MX0 145985242 EC50 = 7.643 nM T44068 C1ZWI5 145986105 EC50 = 35.98 nM T44068 CD62SW 145987168 EC50 = 630.96 nM T44068 C74LVN 145987415 EC50 = 3162.28 nM T44068 CLCV71 145987938 EC50 > 10000 nM T44068 CK1C0A 145989075 EC50 = 831.76 nM T44068 C4GV8Q 145990586 IC50 = 1.7 nM T44068 C0SH3Y 145991661 EC50 > 10000 nM T44068 CT6SD4 145992462 EC50 > 10000 nM T44068 C06QWE 145992510 EC50 > 10000 nM T44068 CV7U8T 145994130 EC50 = 831.76 nM T44068 CC2G1V 146025727 Ki = 8500 nM T44068 CKAW68 146025802 EC50 = 300 nM T44068 CEP41C 146025803 EC50 = 2511.89 nM T44068 C6P3SR 153287553 Ki = 3162.28 nM T44068 CV9G7Z 153287572 Ki > 10000 nM T44068 CO85KL 153287574 Ki > 10000 nM T44068 CB1F6M 155510718 Ki = 1.82 nM T44068 CQ8O2V 155513474 EC50 = 6.761 nM T44068 CQP6N7 155515551 Ki = 1.259 nM T44068 C1N6LR 155515718 EC50 = 1445.44 nM T44068 CP0R2N 155515823 Ki = 83.18 nM T44068 CUM2N4 155515982 Ki = 13000 nM T44068 CERN85 155517986 EC50 = 10000 nM T44068 C8NG9I 155518547 Ki = 44.67 nM T44068 CUSA24 155519891 Ki = 1000 nM T44068 CI5Z4A 155521390 Ki = 269.15 nM T44068 CQL75N 155524038 EC50 = 15.85 nM T44068 CM78EJ 155527605 IC50 = 1778.28 nM T44068 CDJ8F2 155527926 EC50 = 1949.84 nM T44068 CN7D8W 155528927 Ki = 2.884 nM T44068 CABK31 155530927 IC50 = 5.623 nM T44068 CV23QL 155535986 IC50 = 181.97 nM T44068 CB79ZW 155536080 Ki > 10000 nM T44068 C0C1ZH 155536314 EC50 = 218.78 nM T44068 C2GLP7 155536373 Ki = 6.457 nM T44068 CV7X4Y 155536813 EC50 = 11.22 nM T44068 CQY6O9 155537285 Ki = 2570.4 nM T44068 C9U1EQ 155539613 Ki = 1.096 nM T44068 CZ5F4E 155543358 EC50 = 5.012 nM T44068 C62AZC 155543518 EC50 = 239.88 nM T44068 CQK0S7 155544582 Ki = 4.169 nM T44068 C0KO4S 155545790 Ki = 478.63 nM T44068 CAJ01M 155548071 EC50 = 9.772 nM T44068 C17YQR 155550544 EC50 = 15.85 nM T44068 C65JRG 155550964 EC50 = 87.1 nM T44068 CA3ST2 155551006 EC50 = 22.39 nM T44068 C7DE8Z 155551133 EC50 = 72.44 nM T44068 CX8JA1 155552185 Ki > 50000 nM T44068 CTPM05 155557081 IC50 = 4466.84 nM T44068 CB85MA 155557083 EC50 = 36.31 nM T44068 C7EVF6 155559960 Ki = 3.981 nM T44068 CKM05W 155563970 Ki = 19.5 nM T44068 CR8W7Y 155564079 EC50 = 6.31 nM T44068 CL43AX 155564340 EC50 = 13.49 nM T44068 CD78XW 155564766 EC50 = 7.413 nM T44068 CZ51GL 155565922 IC50 = 28.18 nM T44068 CA05IO 155567283 EC50 = 43.65 nM T44068 CMU1C9 155569481 Ki = 8.913 nM T44068 CP9TR0 10324985 Ki = 475.8 nM T44068 CF40LD 44349237 IC50 = 830 nM T44068 CTNO31 44349323 IC50 = 3000 nM T44068 C91AXH 44349356 IC50 = 1800 nM T44068 C9JZ7V 44349357 IC50 = 820 nM T44068 C5TWZ0 44349367 IC50 = 3800 nM T44068 CE2XL3 44349378 IC50 = 1100 nM T44068 C5ELB7 44349379 IC50 = 790 nM T44068 D01JXM 46222048 Ki > 1000 nM T44068 D01OIK 155774 EC50 = 10.96 nM T44068 D02DKX 5311116 EC50 = 2.291 nM T44068 D02VPW 6603756 Ki = 0.25 nM T44068 D03BZW 2687 EC50 = 12.3 nM T44068 D03VHK 10028830 EC50 = 889 nM T44068 D04HXF 4080436 Ki = 12 nM T44068 D05GDP 599482 Ki > 10000 nM T44068 D05JKG 68770 Ki = 240 nM T44068 D05ZUX 44207909 Ki >= 1000 nM T44068 D08BCF 5011 Ki = 6309.57 nM T44068 D09PIN 3378093 Ki > 1000 nM T44068 D09RPR 16737207 Ki > 10000 nM T44068 D0A4FU 2769774 Ki = 114 nM T44068 D0F2SA 46901383 IC50 = 8300 nM T44068 D0J6JT 1355 IC50 = 2000 nM T44068 D0L5MW 181743 Ki = 8565 nM T44068 D0O9HS 415628 IC50 = 12000 nM T44068 D0R3GW 10296414 Ki = 2511.89 nM T44068 D0T2RY 9948320 Ki >= 1000 nM T44068 D0TX8W 594590 Ki = 67.61 nM T44068 D0V4RP 1346 IC50 = 2000 nM T44068 D0X4RC 7096 Ki = 1348.96 nM T59445 D03KOZ 1549120 IC50 = 67700 nM T59445 D0K8KX 5280343 IC50 = 35600 nM T59445 CL70CJ 13650 IC50 = 106000 nM T59445 CA9YN2 99477 IC50 > 400000 nM T59445 CU1EW8 132302 IC50 = 240 nM T59445 CNZ73E 5280567 IC50 = 153000 nM T59445 CRY76T 5319502 IC50 = 212000 nM T59445 C5S4KV 5320203 IC50 = 288000 nM T59445 CFXB53 5338490 IC50 = 163000 nM T59445 CX0I3E 5393159 IC50 = 335000 nM T59445 CWR71Z 9924967 IC50 = 19 nM T59445 CCYD83 9945366 IC50 = 7 nM T59445 CGN2V1 9946410 IC50 = 99 nM T59445 C06EYU 9948799 IC50 = 27 nM T59445 COV86C 9968745 IC50 = 10 nM T59445 C8FX0P 10132209 IC50 = 5 nM T59445 C7YEB6 10133045 IC50 = 130 nM T59445 C2AOX9 10136152 IC50 = 4 nM T59445 CQK30T 10154556 IC50 = 80 nM T59445 CDTY96 10155208 IC50 = 6 nM T59445 CAH3C4 10155331 IC50 = 100 nM T59445 CMC8Y1 10157477 IC50 = 13 nM T59445 C82XRZ 10271780 IC50 = 7 nM T59445 C32HGR 10291693 IC50 = 212 nM T59445 CCX10M 10295175 IC50 = 4 nM T59445 CBW0L7 10869424 IC50 = 1100 nM T59445 CP5EB7 10870950 IC50 = 150 nM T59445 CAM7D5 10872151 IC50 = 67 nM T59445 C3CYE9 10881940 IC50 = 32 nM T59445 CZ1WB8 10890948 IC50 = 9400 nM T59445 C8FYG6 10904343 IC50 = 270 nM T59445 C9GX3J 10912647 IC50 = 2300 nM T59445 CKRC71 10923679 IC50 = 1300 nM T59445 CZ0NH1 10937391 IC50 = 180 nM T59445 CAZU37 10949519 IC50 = 43 nM T59445 C2BF3D 10958350 IC50 = 24 nM T59445 C5R1VI 10969917 IC50 = 490 nM T59445 C3RI4C 10979846 IC50 = 120 nM T59445 CDZR58 10980319 IC50 = 170 nM T59445 CY9V1M 10980854 IC50 = 170 nM T59445 C2CG8Q 10980855 IC50 = 140 nM T59445 CG81SF 10989418 IC50 = 2600 nM T59445 CL5RF2 10991368 IC50 = 4800 nM T59445 C2QPB0 10991473 IC50 = 12 nM T59445 C14ZET 11013235 IC50 = 23 nM T59445 C8IHG4 11015344 IC50 = 190 nM T59445 CYHO07 11035075 IC50 = 36 nM T59445 CYI12F 11035272 IC50 = 80 nM T59445 CV1C7N 11035750 IC50 = 3200 nM T59445 CBV8R0 11045598 IC50 = 35 nM T59445 C16HBP 11046187 IC50 = 200 nM T59445 CI1DO0 11055689 IC50 = 110 nM T59445 C7Z8RC 11056129 IC50 = 31 nM T59445 C10EXV 11056575 IC50 = 486 nM T59445 C1DLS9 11057232 IC50 = 8 nM T59445 CR52FO 11057895 IC50 = 220 nM T59445 CODT41 11067034 IC50 = 173 nM T59445 CDI1B5 11067657 IC50 = 34 nM T59445 CF67SK 11089997 IC50 = 72 nM T59445 CV1NQ8 11099061 IC50 = 23 nM T59445 CL76SF 11099443 IC50 = 80 nM T59445 CM2K1C 11099484 IC50 = 3200 nM T59445 CAO5C9 11109705 IC50 = 190 nM T59445 CBF4N0 11120125 IC50 = 350 nM T59445 C1C8DE 11120462 IC50 = 6500 nM T59445 C6BDJ9 11121071 IC50 = 20 nM T59445 C2B3ZG 11129412 IC50 = 3000 nM T59445 C3LO2X 11130365 IC50 = 140 nM T59445 CBA08V 11141177 IC50 = 260 nM T59445 C3Y9WD 11142000 IC50 = 64 nM T59445 CI6B0K 11727405 IC50 = 44 nM T59445 C26DVI 11761290 IC50 = 120 nM T59445 C4ZNK1 11809438 IC50 = 890 nM T59445 CF1DH4 11823548 IC50 = 37 nM T59445 C48JWY 11834218 IC50 = 590 nM T59445 CA1X7R 22088595 IC50 = 19 nM T59445 CY9WK7 44283102 IC50 = 28 nM T59445 CHA54P 44283319 IC50 = 831 nM T59445 C4DN2E 44366180 IC50 = 40 nM T59445 CDP40Y 44366419 IC50 = 12 nM T59445 C0SC5P 44366420 IC50 = 59 nM T59445 C6NOP2 44366455 IC50 = 10 nM T59445 CAS91K 54682930 IC50 > 400000 nM T59445 D02JEZ 5281426 IC50 = 120000 nM T59445 D03ZMQ 323 IC50 > 400000 nM T59445 D05DAN 9841731 IC50 = 10 nM T59445 D05QOR 5280460 IC50 = 137000 nM T59445 D0E0RW 69894 IC50 > 250000 nM T59445 D0OC4B 5357479 IC50 = 70700 nM T59445 D0U4BB 10748 IC50 = 124000 nM T59445 D0YZ5G 5281416 IC50 = 82900 nM T36741 D0Q7AG 53240420 IC50 = 2000 nM T36741 CN1W8P 1109690 IC50 = 4200 nM T36741 C4TP0I 1109692 IC50 = 630 nM T36741 CV2FP8 1317466 IC50 = 847.4 nM T36741 C0V6NK 2337251 IC50 = 680 nM T36741 CAK8E4 10124724 IC50 = 8000 nM T36741 CDAT72 11433190 IC50 = 4300 nM T36741 CC0E8F 16755649 IC50 > 1000 nM T36741 C5Z6QL 24969086 IC50 = 19700 nM T36741 CQS64F 25105771 IC50 = 22000 nM T36741 C76YPC 44472953 IC50 = 96000 nM T36741 C9F6EY 44472956 IC50 = 41000 nM T36741 CY9G8S 44472957 IC50 = 24000 nM T36741 CU49PM 44472958 IC50 = 36000 nM T36741 CK5U1C 44472959 IC50 = 59000 nM T36741 CA86ZW 44472960 IC50 > 100000 nM T36741 CZ4LN0 44472961 IC50 = 13000 nM T36741 C6MGL0 44472962 IC50 = 20000 nM T36741 CQ84LW 44472963 IC50 = 12000 nM T36741 CG7P3B 44472964 IC50 = 8100 nM T36741 C4CON7 44472965 IC50 = 7500 nM T36741 CPK9V3 44472966 IC50 = 6500 nM T36741 C5BYN0 44472968 IC50 = 10000 nM T36741 C3Z4SR 44472969 IC50 = 8000 nM T36741 C94UNC 44472970 IC50 = 10000 nM T36741 C6HOC3 44472971 IC50 = 4100 nM T36741 CST25L 44472972 IC50 = 7500 nM T36741 C8QNJ9 44472973 IC50 = 2700 nM T36741 CS95EF 44472974 IC50 = 3200 nM T36741 COM24Y 44472975 IC50 = 5100 nM T36741 CNOT62 44472976 IC50 = 14000 nM T36741 C4TI7C 44472977 IC50 = 41000 nM T36741 C5W0VC 44582364 IC50 = 100 nM T36741 C7OYC3 44825260 Ki = 36000 nM T36741 CL68QB 46227513 IC50 > 100000 nM T36741 CZ23MN 52943867 IC50 = 339000 nM T36741 C9Q6TG 52945081 IC50 = 348000 nM T36741 CIQZ61 52945082 IC50 = 463000 nM T36741 CK2V0T 52945083 IC50 = 300000 nM T36741 CJYK89 52947529 IC50 = 192000 nM T36741 C3CV2G 52949945 IC50 = 307000 nM T36741 C59UNR 53317544 IC50 = 340 nM T36741 CC15QU 53317691 IC50 = 1600 nM T36741 C1Q8TB 53318829 IC50 = 1400 nM T36741 CI08RL 53321450 IC50 = 282 nM T36741 C3ML7J 53321451 IC50 = 170 nM T36741 CR90KG 53321452 IC50 = 270 nM T36741 CCV52T 53322772 IC50 = 100 nM T36741 C78AKT 53322773 IC50 = 8300 nM T36741 CTFZ46 53322774 IC50 = 180 nM T36741 CI9H2K 53325414 IC50 = 550 nM T36741 CMT70F 53325415 IC50 = 540 nM T36741 CQ8Y7H 56591370 IC50 > 30000 nM T36741 C62OCN 56951871 IC50 = 19000 nM T36741 C7ZCX9 66561791 IC50 = 18000 nM T36741 CY5W7H 66987552 Ki = 3150 nM T36741 CJD2Q0 70696176 IC50 = 70000 nM T36741 CI6GS5 71305070 IC50 > 30000 nM T36741 COGY08 71305072 IC50 > 30000 nM T36741 C60FEX 71544420 IC50 > 100000 nM T36741 CC9H1S 71585475 IC50 = 4160 nM T36741 CBLH41 71663696 IC50 > 30000 nM T36741 CI4ZS6 71678942 IC50 = 27800 nM T36741 CKC91P 72714997 IC50 = 42100 nM T36741 CN75KD 72714998 IC50 = 52500 nM T36741 CG5X1Q 73347121 IC50 = 1128 nM T36741 CME7R0 73348988 IC50 = 32400 nM T36741 C7XN3A 73386675 IC50 > 100000 nM T36741 CNB31V 86766851 IC50 = 468 nM T36741 CKA25D 90666824 IC50 = 13000 nM T36741 CKGW70 90666826 IC50 = 7000 nM T36741 CE89VR 90666827 IC50 = 900 nM T36741 C7FKE1 90666833 IC50 > 50000 nM T36741 C3Z8WE 90666834 IC50 > 50000 nM T36741 C03GLI 90666835 IC50 = 30000 nM T36741 CE5FT8 90666836 IC50 = 30000 nM T36741 CL9H7W 90666837 IC50 = 42000 nM T36741 CP5GD7 90666838 IC50 > 50000 nM T36741 CLA53P 90666839 IC50 = 963000 nM T36741 CU91QC 90666840 IC50 = 1684000 nM T36741 C5W9VY 90666841 IC50 = 3486000 nM T36741 CPJ8A5 90666842 IC50 = 3428000 nM T36741 CLV12D 90667000 IC50 = 4916000 nM T36741 C82EPU 90667001 IC50 = 5322000 nM T36741 C0FG5C 90667002 IC50 = 20000 nM T36741 CC3FL7 118718047 IC50 = 1650 nM T36741 CNQT35 118718079 Ki > 50000000 nM T36741 CFHE72 122689625 IC50 = 140 nM T36741 C95MAK 126963310 Ki = 26300 nM T36741 C6I9MQ 127035023 Ki > 60000 nM T36741 CSI49A 127035024 Ki > 60000 nM T36741 CD0Q5H 127035025 Ki > 60000 nM T36741 CFZ35L 127035026 Ki = 5000 nM T36741 CFK31G 127035027 Ki = 200 nM T36741 CVY7S6 127035701 Ki = 1500 nM T36741 CF86ES 127035702 Ki = 6090 nM T36741 C68JWY 136209736 IC50 = 25 nM T36741 C3ZGV0 137631366 Ki = 4170 nM T36741 CC3HQ7 137633155 IC50 = 4.6 nM T36741 CWY4X0 137633285 IC50 = 3.3 nM T36741 CGHT40 137633360 Ki = 6990 nM T36741 CZ31RB 137637908 IC50 = 55.8 nM T36741 CP1HD6 137639153 Ki = 14700 nM T36741 C17SXB 137640724 IC50 = 207.4 nM T36741 CQ8P1F 137642328 Ki = 4400 nM T36741 CC13NQ 137644080 Ki = 44000 nM T36741 C1TYP0 137645068 Ki = 55000 nM T36741 C0WHG9 137645614 Ki = 35300 nM T36741 C61JDO 137646640 IC50 = 22.8 nM T36741 CQLA87 137647053 Ki = 9750 nM T36741 C43INM 137647313 IC50 = 214.5 nM T36741 CUL1O6 137647880 Ki = 4290 nM T36741 CE3V8Y 137650518 Ki = 40200 nM T36741 C7KZ4L 137653948 IC50 = 401 nM T36741 C2OJU7 137654973 Ki = 27400 nM T36741 CIC2K9 137655254 Ki = 4710 nM T36741 C8R0UO 137655459 IC50 = 10.7 nM T36741 C4HB1U 137656155 IC50 = 6.1 nM T36741 C2QHP5 137656534 IC50 = 10.4 nM T36741 CU3FN6 137657022 IC50 = 136.4 nM T36741 CPHT95 137657789 Ki = 6760 nM T36741 C7QF5S 137658136 Ki = 12400 nM T36741 CTM69S 137658613 Ki = 46000 nM T36741 CDMY96 137659576 IC50 = 87.9 nM T36741 C3JM5Y 137660704 Ki = 29600 nM T36741 CHD18T 137661621 Ki = 4910 nM T36741 CWJ84Q 137662288 Ki = 16170 nM T36741 C0X8ER 145949722 IC50 > 1000 nM T36741 C2MO7K 145951845 IC50 > 1000 nM T36741 CG80FB 145951878 IC50 = 302 nM T36741 C1P0NL 145952828 IC50 = 77.4 nM T36741 CJA7N9 145953608 IC50 > 1000 nM T36741 CZ4SK6 145954275 IC50 > 1000 nM T36741 CTA08K 145956036 IC50 = 57.5 nM T36741 CY5I1O 145956101 IC50 = 12.1 nM T36741 C8RAG3 145956154 IC50 > 1000 nM T36741 CCB51L 145956802 IC50 > 1000 nM T36741 CTS5R3 145959048 IC50 = 219 nM T36741 CQ4ET5 145959752 IC50 = 836 nM T36741 CO0W4J 145961652 IC50 = 81.9 nM T36741 C23HZY 145971531 IC50 = 812 nM T36741 C7DSC3 145980812 Ki = 1400 nM T36741 CW7ZU8 145982231 Ki = 2200 nM T36741 CVEW14 145987298 Ki = 490 nM T36741 CO41YV 145991230 Ki = 2100 nM T36741 CNH2T4 145992205 Ki = 4200 nM T36741 CPF13W 145993071 Ki = 2600 nM T36741 CG5FX7 155515298 IC50 = 3600 nM T36741 CWI45U 155517444 Ki = 8060 nM T36741 CNGH35 155521620 Ki = 12600 nM T36741 CZ21FA 155522131 Ki = 5450 nM T36741 CCX4D5 155522186 Ki = 8010 nM T36741 CB8G5R 155523298 Ki = 5740 nM T36741 C78PNX 155523379 Ki = 6390 nM T36741 C0HAV7 155524001 Ki = 4740 nM T36741 C7N0SY 155526905 Ki = 8640 nM T36741 CJC07B 155527872 IC50 = 7100 nM T36741 CI16PB 155528357 IC50 = 4900 nM T36741 CWC32Z 155529926 Ki = 20500 nM T36741 C5R8YO 155530377 Ki = 3630 nM T36741 CYL1M7 155532432 Ki = 11150 nM T36741 CKUT47 155534630 Ki = 1550 nM T36741 CWGE76 155537056 IC50 = 6600 nM T36741 CJ9SV2 155539377 IC50 = 2.1 nM T36741 C9T2LU 155539551 Ki = 4670 nM T36741 CZJ43Y 155540256 Ki = 6300 nM T36741 C5BLH7 155541232 IC50 = 3900 nM T36741 C4E6YV 155541314 Ki = 7050 nM T36741 CS74BO 155541655 Ki = 6010 nM T36741 C7DH4S 155542925 IC50 = 6000 nM T36741 CYXP56 155543879 IC50 = 7600 nM T36741 CUS85I 155546101 IC50 = 5000 nM T36741 CVG09H 155546326 Ki = 1950 nM T36741 CD54OX 155546509 Ki = 4010 nM T36741 CV76YM 155547556 Ki = 4730 nM T36741 CW8J1M 155548484 Ki = 6030 nM T36741 C7E9DQ 155550524 Ki = 5780 nM T36741 CC5LD1 155554511 Ki = 3960 nM T36741 CKOD46 155554714 Ki = 15740 nM T36741 CMI3L2 155555639 Ki = 1680 nM T36741 C7ZF4U 155558272 Ki = 7250 nM T36741 C7YWV8 155558664 Ki = 5360 nM T36741 C0PR4Z 155558699 Ki = 6760 nM T36741 CSER69 155561097 Ki = 20900 nM T36741 CUE2F7 155564869 Ki = 6210 nM T36741 C5IBV6 155565604 Ki = 4740 nM T36741 C3QM1J 155568384 Ki = 6380 nM T36741 C5D8PE 155569182 IC50 = 16600 nM T36741 C8KE3W 155569673 Ki = 6840 nM T36741 D01QKK 216345 IC50 > 10000 nM T44916 D00EQL 66558664 IC50 = 2 nM T44916 D0Y2HR 2247 Ki = 23010 nM T44916 CSH9X6 114551 IC50 > 500000 nM T44916 CW4O3G 3818672 IC50 > 500000 nM T44916 C53MPU 5005916 IC50 = 146000 nM T44916 C0AXH6 10015659 IC50 = 6040 nM T44916 C7Y8BE 17039514 IC50 = 95000 nM T44916 CY84LN 29111296 IC50 = 620 nM T44916 C4G5LK 31301024 Ki = 1500 nM T44916 C37ZXI 84784098 IC50 = 95000 nM T44916 C4RV3D 84784100 IC50 = 40000 nM T44916 C3NPY4 84786790 IC50 = 35000 nM T44916 C29CSY 84789118 IC50 = 119000 nM T44916 CI68GL 95854752 Ki = 1500 nM T44916 CBZU50 118996396 IC50 > 100000 nM T44916 C42XHL 123132213 Ki = 0.3 nM T44916 CE4J7X 123132216 Ki = 1 nM T44916 CYJX49 123132228 IC50 = 220 nM T44916 CXHL60 123132930 IC50 = 1650 nM T44916 CYX90I 124037093 Ki = 600 nM T44916 CEM89S 124220775 Ki = 2.6 nM T44916 C0LO1N 124220776 Ki = 10 nM T44916 C6WF0P 126962003 Ki = 4 nM T44916 CMBD89 132085494 Ki = 0.29 nM T44916 C3AZ4U 132085564 Ki = 129 nM T44916 CP5VY8 132085570 Ki = 0.45 nM T44916 CT4D7X 132085601 Ki = 18 nM T44916 C1ZTP9 132085608 Ki = 0.3 nM T44916 CJEB10 132085621 Ki = 3 nM T44916 CN2VX7 132085691 Ki = 42 nM T44916 CQ4V0M 137349702 IC50 = 2500 nM T44916 C91XMO 137349703 IC50 = 1000 nM T44916 C0U4VB 137631567 IC50 = 70 nM T44916 CK9DX7 137631625 IC50 = 150 nM T44916 CEV81K 137631673 Ki = 0.74 nM T44916 CR5NJ9 137631817 IC50 = 80 nM T44916 C0HSD4 137631902 IC50 = 49 nM T44916 CHKA43 137632081 IC50 = 290 nM T44916 CD39VC 137632104 IC50 = 130 nM T44916 C0L5KQ 137632213 IC50 = 510 nM T44916 C1V0GR 137632262 IC50 = 80 nM T44916 C6XIK0 137632301 IC50 = 62 nM T44916 CX2M8L 137632658 Ki = 80 nM T44916 C3RKW2 137632692 IC50 = 290 nM T44916 CA2S4D 137633269 IC50 = 110 nM T44916 C1JG7S 137633327 Ki = 49 nM T44916 CI9ZT5 137633377 IC50 = 1000 nM T44916 CV01UF 137633485 Ki = 23 nM T44916 COG6Y5 137633952 IC50 = 60 nM T44916 CUB38O 137634105 IC50 = 180 nM T44916 C2YJ3D 137634224 IC50 = 80 nM T44916 C3AS8E 137634542 IC50 = 2180 nM T44916 CR3T6Y 137635115 IC50 = 70 nM T44916 CL7NQ2 137635373 IC50 = 21800 nM T44916 C1I5KT 137636203 Ki = 66 nM T44916 CYA4D2 137636441 IC50 = 120 nM T44916 CD86SJ 137636483 Ki > 50000 nM T44916 CIC97Z 137636493 IC50 = 30 nM T44916 CX3D9A 137636503 Ki = 680 nM T44916 CMN6U1 137637446 IC50 = 160 nM T44916 C97DYW 137637590 IC50 = 440 nM T44916 C6FZ9O 137637638 IC50 = 2340 nM T44916 C4T2LW 137637933 Ki = 2.1 nM T44916 CCG3R6 137638056 IC50 = 50 nM T44916 CDX5U2 137638712 Ki = 10 nM T44916 CV6M3S 137639502 Ki = 4.6 nM T44916 CG3W0R 137639788 IC50 = 40 nM T44916 CP34MJ 137639984 IC50 = 260 nM T44916 CPH8Z0 137640410 IC50 = 80 nM T44916 CA7F2D 137640439 Ki = 260 nM T44916 C9DCO5 137640714 IC50 = 70 nM T44916 CMD73K 137641043 Ki = 0.65 nM T44916 CL02JS 137641418 Ki = 18 nM T44916 C1AUW3 137641587 Ki = 45 nM T44916 C8NIH4 137641805 Ki > 50000 nM T44916 CT26GQ 137642207 IC50 = 40 nM T44916 C10HUF 137642235 IC50 = 2220 nM T44916 CXRJ80 137642432 IC50 = 174000 nM T44916 C3U8IW 137642523 IC50 = 9 nM T44916 C1R4NA 137642569 IC50 = 160 nM T44916 CWLE27 137642570 IC50 = 3520 nM T44916 CU76BI 137643206 IC50 = 80 nM T44916 C8MG4Z 137643251 IC50 = 90 nM T44916 CA04WV 137643374 IC50 = 130 nM T44916 CD9J8L 137643872 Ki = 71 nM T44916 CV40XW 137643933 IC50 = 1300 nM T44916 C4N2JQ 137644092 Ki = 230 nM T44916 CY2A7B 137644185 IC50 = 43000 nM T44916 C80NXA 137644277 IC50 = 170 nM T44916 C6S3PQ 137644620 IC50 = 150 nM T44916 C0WHJ4 137645378 IC50 = 270 nM T44916 C30QAS 137645890 IC50 = 140 nM T44916 C0QO5D 137645987 IC50 = 20 nM T44916 CADX27 137646001 Ki > 50000 nM T44916 CRB91Z 137646136 IC50 = 310 nM T44916 C61END 137646227 IC50 = 13 nM T44916 CZ7JE1 137646443 Ki = 2.6 nM T44916 CI7QO6 137646599 Ki = 78 nM T44916 CZ9R4P 137646792 Ki = 78 nM T44916 C0ZAK8 137646810 IC50 = 94 nM T44916 C5OD2A 137647698 IC50 = 110 nM T44916 C62GUF 137648098 IC50 = 53 nM T44916 CTHZ72 137648271 IC50 = 50 nM T44916 C4O7UA 137648303 IC50 = 20490 nM T44916 CGW83R 137648968 IC50 = 21800 nM T44916 C9AK1N 137649814 IC50 = 2500 nM T44916 CUB7S5 137650115 IC50 = 70 nM T44916 C96FDA 137650497 Ki = 5.3 nM T44916 CW81FV 137650740 Ki = 1 nM T44916 CXGT40 137650766 Ki = 12 nM T44916 C0C4TZ 137650804 Ki = 56 nM T44916 C2AL4I 137650810 IC50 = 9 nM T44916 C23WLV 137651012 IC50 = 770 nM T44916 C5OV6C 137651308 IC50 = 10 nM T44916 CMT0P2 137651353 IC50 = 2700 nM T44916 CDN27H 137651601 IC50 = 70 nM T44916 CWI0T7 137651727 Ki = 18 nM T44916 CHVX90 137651882 IC50 = 49 nM T44916 C5YLC4 137651932 IC50 = 160 nM T44916 CMHQ27 137652034 IC50 = 7900 nM T44916 CA85WK 137653282 IC50 = 20 nM T44916 C8IJ0W 137653495 Ki = 450 nM T44916 CC3O1L 137654064 IC50 = 69 nM T44916 CX47EU 137654124 IC50 = 90 nM T44916 C78XUM 137654221 IC50 = 30 nM T44916 CAW9N1 137654472 Ki = 290 nM T44916 C20VKL 137654491 IC50 = 40 nM T44916 CG3B9Z 137655015 Ki = 53 nM T44916 CP82UT 137655616 Ki = 0.3 nM T44916 CB3ST5 137655692 IC50 = 70 nM T44916 C1IF3D 137656070 IC50 = 30 nM T44916 CJX16G 137656135 IC50 = 30 nM T44916 CN42VT 137656162 IC50 = 2100 nM T44916 CQ0B5W 137656316 IC50 = 100 nM T44916 C7SE6J 137656811 IC50 = 150 nM T44916 C4P0NB 137656935 IC50 = 1600 nM T44916 C2V1EB 137657094 Ki = 160 nM T44916 C1M9WN 137657139 IC50 = 19 nM T44916 CYHA48 137657149 IC50 = 30 nM T44916 CSH38D 137657176 IC50 = 69 nM T44916 CU8V6M 137657184 Ki = 91 nM T44916 C9VI4T 137657192 IC50 = 260 nM T44916 CK7E2L 137657380 IC50 = 52 nM T44916 C2K4HB 137657595 IC50 = 7 nM T44916 CJG53C 137657817 Ki > 50000 nM T44916 C8SY3I 137658035 Ki = 59 nM T44916 C86YUI 137658285 IC50 = 130 nM T44916 CBR2P4 137658502 Ki = 330 nM T44916 CX86QR 137658665 IC50 = 80 nM T44916 C1LFE3 137659068 Ki = 610 nM T44916 CH86OM 137659179 Ki = 3 nM T44916 COVX53 137659190 IC50 = 12400 nM T44916 CIK1U5 137659343 IC50 = 110 nM T44916 CPM13C 137659477 IC50 = 90 nM T44916 CN6QM1 137660778 IC50 = 14900 nM T44916 C84DXZ 137660820 IC50 = 2000 nM T44916 CXW54U 137661084 IC50 = 40 nM T44916 C7K4CA 137661104 IC50 = 93 nM T44916 C52XHW 137661318 IC50 = 14080 nM T44916 CET87X 137661547 Ki = 380 nM T44916 C1MZG7 137661702 Ki = 8 nM T44916 C4FR5B 137661879 IC50 = 20 nM T44916 C10TSN 145950077 IC50 = 1740 nM T44916 CM0VX9 145958430 IC50 = 3870 nM T44916 D0B4DP 9877750 Ki = 950 nM T33211 D02TJS 54676038 IC50 = 1300 nM T33211 D0E3OF 54678486 IC50 = 24590 nM T33211 CUS16Z 44584846 Ki = 135 nM T33211 CP2J8X 44584953 Ki = 206 nM T33211 CBX8K0 44584960 Ki = 172 nM T33211 C10KCB 44584961 Ki = 1133 nM T33211 C1S6KQ 44584962 Ki = 1220 nM T33211 CJ73BT 45486346 Ki > 10000 nM T33211 C9ETC4 45486354 Ki > 10000 nM T33211 CVPG40 45486356 Ki = 968 nM T33211 CSQ2K4 45486357 Ki = 5131 nM T33211 CX2FT3 53344593 IC50 = 462 nM T33211 CJ2W9V 75593418 Ki = 72 nM T33211 C0ET8W 137630787 Ki = 0.12 nM T33211 D05JJL 44584947 Ki = 135 nM T33211 D0A6FZ 75593419 Ki = 13.8 nM T33211 D0Y9PH 45486355 Ki = 6154 nM T78543 D0E3TC 44259 IC50 = 1.23 nM T78543 D0I4TH 24788740 IC50 = 69 nM T78543 D0MS3Z 16725726 IC50 = 33 nM T78543 D03BNU 59604787 IC50 > 10000 nM T78543 D0T3ME 156422 IC50 > 30000 nM T78543 C6XY0Z 10133248 IC50 > 1000 nM T78543 C54YXC 16121514 IC50 = 41.69 nM T78543 C5VPH9 16129448 IC50 > 10000 nM T78543 C0B7RT 25057409 IC50 = 5600 nM T78543 CSI0U1 44819541 IC50 = 3000 nM T78543 CX6PZ9 51003130 IC50 = 1 nM T78543 C8NA4L 53384644 IC50 > 30000 nM T78543 CV63UL 67240318 IC50 > 10000 nM T78543 C5D1LV 70687790 IC50 = 1862.09 nM T78543 CI1E8V 137634241 IC50 > 10000 nM T78543 C2MD1Q 155513187 IC50 = 517 nM T78543 C41XDM 155537557 IC50 > 1000 nM T98698 D0E3SH 6918837 Ki = 2.3 nM T98698 D0E7PQ 5311 IC50 = 34 nM T98698 D0L7LC 5352062 Ki = 1250 nM T98698 D0Y3KG 3121 IC50 > 2000000 nM T98698 D00FHR 9865515 IC50 > 10000 nM T98698 D05KED 53340666 IC50 = 1400 nM T98698 D09XIZ 11538455 Ki = 1.7 nM T98698 D0B3FV 6445533 IC50 = 2240 nM T98698 D0B7CH 4775 IC50 > 2000000 nM T98698 D0E6UZ 54575456 IC50 = 27 nM T98698 D0GE5B 56654642 IC50 > 180000 nM T98698 D0GH3Q 9804992 Ki = 240 nM T98698 D0L2UQ 49855250 Ki = 107 nM T98698 D0M8FD 4261 IC50 > 1000 nM T98698 D0XT6W 6918638 Ki = 51 nM T98698 D0Z4RC 24756910 IC50 = 373 nM T98698 D0J8OC 5186 IC50 = 2100 nM T98698 D00HXJ 118884610 Ki = 442 nM T98698 D0CH8Q 56965342 IC50 = 4100 nM T98698 D0L1NO 72722126 IC50 = 30 nM T98698 D0QX3G 71532921 IC50 > 10000 nM T98698 D0YN2T 86302836 IC50 = 23 nM T98698 CBIR94 10313 IC50 = 15600 nM T98698 C1N2KZ 88129 IC50 = 99000 nM T98698 C35INR 338818 IC50 = 16160 nM T98698 CH1JD3 419176 IC50 > 1000000 nM T98698 CU3HS2 1108280 IC50 > 100000 nM T98698 C1RD7E 6918878 IC50 > 10000 nM T98698 CE9LP2 9543539 IC50 > 180000 nM T98698 CJ84NF 9815304 IC50 > 10000 nM T98698 CC0EU7 9828788 IC50 = 1760 nM T98698 C81EYJ 9923508 IC50 = 6.3 nM T98698 CL4C9H 10154438 Ki = 324.7 nM T98698 C7RC1E 10309899 IC50 = 46 nM T98698 CG9L1R 10435243 IC50 = 785.9 nM T98698 C60QVT 10460379 IC50 = 1293 nM T98698 CRZ7H2 11556677 IC50 > 10000 nM T98698 CQ32FV 11664499 IC50 = 4200 nM T98698 CG9OC4 11682502 IC50 = 102 nM T98698 CYB26W 11688197 IC50 > 1000 nM T98698 CC3GQ0 11700059 IC50 > 10000 nM T98698 C9G1BN 11993595 IC50 = 4200 nM T98698 CH5JS7 11993694 IC50 = 420 nM T98698 CXJ5G9 13190582 IC50 > 10000 nM T98698 C06UTF 13507024 IC50 = 980 nM T98698 C1KR4L 14113324 IC50 > 50000 nM T98698 C2D1KP 15983982 Ki = 70 nM T98698 CHB82E 15986417 IC50 = 75100 nM T98698 C52EVH 15986418 IC50 = 15600 nM T98698 CS1QO9 15986509 IC50 = 213000 nM T98698 CM3T2E 16049824 IC50 > 1 nM T98698 CFK8J5 16068056 Ki = 89 nM T98698 CMQP70 16068495 Ki = 77 nM T98698 CT84XO 16068594 Ki = 41 nM T98698 CF3ZG5 16068595 Ki = 35 nM T98698 CL60CA 16068912 Ki = 42 nM T98698 C5CIB4 16663079 IC50 > 50000 nM T98698 CWO7V0 16733295 IC50 = 1290 nM T98698 CV54SY 16733414 IC50 = 2780 nM T98698 C8RC9P 24744325 IC50 > 50000 nM T98698 C17GDO 24779722 IC50 = 432 nM T98698 CIO7Q6 24853792 IC50 > 10000 nM T98698 CBN0J5 24853793 IC50 > 1 nM T98698 CV8EF6 25032862 IC50 > 50000 nM T98698 CX69SY 25066355 IC50 = 1720 nM T98698 CF8VP4 25066356 IC50 = 738 nM T98698 CS9XH7 25066547 IC50 = 764 nM T98698 C46AGN 25066548 IC50 = 72.6 nM T98698 CJF2M7 25066549 IC50 = 279 nM T98698 C4I1CJ 25155417 IC50 > 30000 nM T98698 CB4E2J 25155956 IC50 > 50000 nM T98698 CO14XG 25195084 IC50 > 20000 nM T98698 CCD5M7 25227504 IC50 = 27.8 nM T98698 CK0D5S 25227505 IC50 = 180 nM T98698 CN97JP 25227508 IC50 = 61.2 nM T98698 CW8R1B 25227513 IC50 = 271 nM T98698 C43BHY 25269097 IC50 = 1500 nM T98698 C2LES7 42599455 IC50 = 4.4 nM T98698 C2KO0F 42599456 IC50 = 3 nM T98698 C1UAO7 42601485 IC50 > 50000 nM T98698 CDT65Y 42631047 IC50 > 100000 nM T98698 CO57GS 44138033 IC50 = 36300 nM T98698 C5VP4D 44454144 IC50 > 50000 nM T98698 C7F8YJ 44543715 Ki = 7000 nM T98698 CEM91G 44562802 IC50 = 70 nM T98698 C7DS4E 44585337 IC50 = 18700 nM T98698 CA6Q9Y 44592060 IC50 = 22300 nM T98698 C5H8RA 44598536 IC50 > 10000 nM T98698 CC2QV9 44623002 IC50 > 50000 nM T98698 CVJ51M 44623152 IC50 > 50000 nM T98698 C6TJ2G 44623153 IC50 > 50000 nM T98698 CO7S9W 44626297 IC50 = 110 nM T98698 C96ROY 45482635 IC50 > 10000 nM T98698 CV74KP 45482658 IC50 > 10000 nM T98698 CHC0Y1 45482667 IC50 = 350 nM T98698 C90NYX 46896338 IC50 > 30000 nM T98698 CL7PS1 49831258 IC50 > 50000 nM T98698 CI5L2P 49846123 IC50 = 67064.24 nM T98698 C4DL0M 49847150 IC50 = 3720 nM T98698 CC7Y9U 49850262 IC50 = 379 nM T98698 C50PXU 49855444 IC50 > 50000 nM T98698 C78GKN 53361474 IC50 = 4510 nM T98698 CNB63X 53361475 IC50 = 2230 nM T98698 CQ43VH 53363518 Ki = 12 nM T98698 C6Y2EV 53374826 IC50 > 100000 nM T98698 CYQV72 54030066 IC50 = 70 nM T98698 C5A7MU 54613496 IC50 = 313 nM T98698 C7OJ4K 56602459 IC50 > 50000 nM T98698 CSY2L7 56602461 IC50 = 11000 nM T98698 CIO96M 56659403 IC50 > 100000 nM T98698 CL18NI 56666337 IC50 > 100000 nM T98698 C9LC5Y 56673234 IC50 > 100000 nM T98698 CWH5N4 56673261 IC50 > 100000 nM T98698 C0ZJG3 56676500 IC50 = 27000 nM T98698 CFUT54 56682413 IC50 = 24000 nM T98698 CZ25SN 56935695 IC50 > 30000 nM T98698 CG6Z2X 57326710 IC50 = 45000 nM T98698 C10DMC 57336560 Ki = 2500 nM T98698 C4LI0D 57521296 IC50 = 20 nM T98698 CA5Q6O 58147189 IC50 > 50000 nM T98698 C4DYC0 58147224 IC50 > 50000 nM T98698 CMP04X 58147302 IC50 > 50000 nM T98698 CLD40J 58465708 IC50 = 35000 nM T98698 C1MB4Q 59323957 IC50 > 30000 nM T98698 CK6LX0 59454220 IC50 > 30000 nM T98698 C2SDN1 59454252 IC50 > 30000 nM T98698 CO6A2S 59585196 IC50 = 29000 nM T98698 CPZ5Q3 60148646 IC50 = 460 nM T98698 CP2HK9 60148667 IC50 = 120 nM T98698 C8ZL3J 60148690 IC50 = 60 nM T98698 CK5N4E 60148693 IC50 = 30 nM T98698 C27DKW 60148711 IC50 = 110 nM T98698 CS2E6C 60148712 IC50 = 220 nM T98698 CPF50R 60148997 IC50 = 1100 nM T98698 CB7X2E 60151224 IC50 > 10000 nM T98698 CY05OU 60151225 IC50 > 10000 nM T98698 CWO8H0 60152596 IC50 > 10000 nM T98698 CBN3L0 69950064 Ki = 39 nM T98698 CQY1I6 70789579 Ki = 3940 nM T98698 CKR6U8 71583101 IC50 = 200 nM T98698 CBZ5S9 71583103 IC50 = 100 nM T98698 C3PSJ9 71583105 IC50 = 100 nM T98698 C7HG0K 71655802 IC50 = 12610 nM T98698 CPJ4V7 71680913 IC50 = 13000 nM T98698 CI9G3B 71681069 IC50 = 8400 nM T98698 CFUC24 71722010 IC50 > 10000 nM T98698 CI9H6L 72164895 IC50 = 13220 nM T98698 C6RI4C 72195326 IC50 = 7980 nM T98698 CA8D1R 72195458 IC50 = 12680 nM T98698 C0DR7G 72195459 IC50 = 4490 nM T98698 CFK2Z7 72195460 IC50 = 5600 nM T98698 CNJ8X0 72195461 IC50 = 854 nM T98698 CV13FT 72195463 IC50 = 1460 nM T98698 CVXZ50 72195464 IC50 = 355 nM T98698 CM41HG 72195593 IC50 = 360 nM T98698 C5X2IY 72195594 IC50 = 311 nM T98698 C3N8UH 72195595 IC50 = 628 nM T98698 C3WQV2 72375562 IC50 = 960 nM T98698 CV09DJ 72734543 IC50 > 10000 nM T98698 CX3W1T 73333311 IC50 = 4600 nM T98698 CM6H9C 76324878 IC50 = 10 nM T98698 CKI74A 76853213 IC50 > 20000 nM T98698 CJ6Z0X 78324068 IC50 > 20000 nM T98698 C3U0KE 81689842 IC50 = 31 nM T98698 C61VCD 86294741 IC50 = 50000 nM T98698 CBWV30 86294747 IC50 = 49000 nM T98698 C06YBD 86302594 IC50 = 2510 nM T98698 C6M9PL 86765212 IC50 = 4110 nM T98698 CS5I4Y 87261507 IC50 = 290 nM T98698 CYW51P 90654946 IC50 = 49200 nM T98698 CJH1S6 90654947 IC50 = 77200 nM T98698 CSR56C 90655296 IC50 = 45500 nM T98698 CSDO81 90664458 Ki = 104 nM T98698 C0RX4B 90667452 IC50 = 14130 nM T98698 C8HL5V 90667453 IC50 = 22910 nM T98698 C3IE7F 90667454 IC50 = 690 nM T98698 C37GOB 90667455 IC50 = 10720 nM T98698 CJO6T1 91810840 IC50 = 1100 nM T98698 C34WIG 92045024 IC50 = 30800 nM T98698 C9OC0F 101882265 IC50 = 60700 nM T98698 CSU52M 118656852 IC50 = 200 nM T98698 CB6AJ9 118656853 IC50 = 100 nM T98698 CW3Y7E 118714368 IC50 = 7940 nM T98698 CM27KC 118714374 IC50 = 2920 nM T98698 C86WSR 118714378 IC50 = 960 nM T98698 C2W0KJ 118714380 IC50 = 7680 nM T98698 CL3ZF9 118714381 IC50 = 770 nM T98698 CMJF26 118714382 IC50 = 4400 nM T98698 CV04TX 118714383 IC50 = 530 nM T98698 C8LVO5 118714384 IC50 = 487 nM T98698 CI8G4X 118737400 IC50 = 8770 nM T98698 C9S5OK 121279020 IC50 > 50000 nM T98698 CIA40K 121472983 IC50 > 10000 nM T98698 CL3M2F 121499152 IC50 > 33330 nM T98698 C28JVO 122192004 IC50 > 10000 nM T98698 CF2D8U 122192005 IC50 > 10000 nM T98698 C3V5ND 122550211 IC50 > 10000 nM T98698 CZE35C 122648343 IC50 > 1000 nM T98698 C54RNT 122648367 IC50 > 1000 nM T98698 C1UVI7 122648600 IC50 > 1000 nM T98698 CMX59K 122648648 IC50 = 650 nM T98698 CVZ64I 122648649 IC50 = 895 nM T98698 CV9I8D 127030313 IC50 = 10900 nM T98698 CB8HR2 129104138 IC50 = 3400 nM T98698 CCH65A 129104183 IC50 > 50000 nM T98698 CFH8Q4 129104227 IC50 > 50000 nM T98698 C6HM5P 129104349 IC50 > 50000 nM T98698 CZTF90 129104374 IC50 > 50000 nM T98698 CUJ2P5 129104402 IC50 > 50000 nM T98698 C6X3HG 132145728 IC50 = 766 nM T98698 C8O9DP 132157820 IC50 = 709 nM T98698 C05FVT 134492522 IC50 > 10000 nM T98698 C14FWK 135348858 IC50 = 8340 nM T98698 CS1V6A 135367138 IC50 > 50000 nM T98698 CVO59N 135367789 IC50 > 50000 nM T98698 CDY18W 135407493 IC50 > 100000 nM T98698 CW2I4R 135412048 IC50 > 100000 nM T98698 C7U0AV 135412194 IC50 > 100000 nM T98698 CS54TL 135437514 IC50 > 100000 nM T98698 C36MUC 135441620 IC50 > 100000 nM T98698 CRB8M1 135444536 IC50 > 100000 nM T98698 CX5D6J 135446479 IC50 = 24400 nM T98698 C1TOK2 135449197 IC50 > 100000 nM T98698 CW25GL 135462117 IC50 > 100000 nM T98698 CCL28F 135473106 IC50 > 100000 nM T98698 CYA60G 135497781 IC50 > 100000 nM T98698 C8X5LO 135928012 Ki = 1100 nM T98698 CI2YE8 135928628 IC50 > 100000 nM T98698 C50NIS 136025837 IC50 > 100000 nM T98698 C4OS0V 136025842 IC50 > 100000 nM T98698 CX7Z5B 136025843 IC50 > 100000 nM T98698 CB8EM9 136025984 IC50 > 100000 nM T98698 C49MUG 136025986 IC50 > 100000 nM T98698 CH7Y3C 136086920 IC50 > 100000 nM T98698 C3VDL5 136086921 IC50 > 100000 nM T98698 C9GOB5 136086922 IC50 > 100000 nM T98698 CE3ZL7 136086923 IC50 > 100000 nM T98698 CJZ5F3 136086924 IC50 = 31900 nM T98698 CT19ND 136110961 IC50 > 100000 nM T98698 CY9U0E 136173089 IC50 > 50000 nM T98698 C67EFJ 137628684 IC50 > 1000 nM T98698 CP0BN3 137631704 Ki > 50000 nM T98698 CZ1FK2 137635119 IC50 > 50000 nM T98698 C6JVG9 137635398 IC50 = 17200 nM T98698 CGMN16 137647616 Ki > 50000 nM T98698 CDXE54 137649646 Ki > 50000 nM T98698 C5FHD3 137652442 IC50 = 30 nM T98698 CB15PI 137652670 Ki > 50000 nM T98698 C1SBN5 137654946 IC50 = 958 nM T98698 CI6R3W 137656303 Ki > 50000 nM T98698 C76OGQ 137656942 IC50 = 22000 nM T98698 C1DL3P 137657892 Ki > 50000 nM T98698 C8D2GT 137658785 Ki > 50000 nM T98698 CAQ62X 137701235 Ki = 1700 nM T98698 CN2UH1 139303146 IC50 > 20000 nM T98698 C7XI0V 141764754 IC50 = 392 nM T98698 CKBF56 142506033 IC50 = 90810 nM T98698 CGNQ74 142506189 IC50 = 229 nM T98698 C1T3IQ 142506210 IC50 = 24400 nM T98698 CEGV67 142506220 IC50 = 23120 nM T98698 CP5HF8 142506225 IC50 = 60 nM T98698 CV3QO5 145951170 IC50 > 10000 nM T98698 CKG98W 145953085 IC50 > 100000 nM T98698 C9IV1C 145959866 IC50 > 10000 nM T98698 CK1XI0 145960971 IC50 > 10000 nM T98698 CP53JS 145977717 IC50 > 10000 nM T98698 CWD0A9 145983712 Ki > 10000 nM T98698 C56MWZ 145986208 Ki > 10000 nM T98698 C0GMR1 146585718 IC50 = 104 nM T98698 C0YXS8 147254231 IC50 = 10410 nM T98698 CN71OS 149405396 IC50 > 100000 nM T98698 C8S3MF 150076000 IC50 > 300 nM T98698 CWG10H 151364732 IC50 > 10000 nM T98698 C6I7OZ 152636346 IC50 > 10000 nM T98698 C7LM4U 153534003 IC50 > 10000 nM T98698 CP1V9H 153534004 IC50 > 10000 nM T98698 C9FIY4 153534005 IC50 > 10000 nM T98698 CVT63S 153534008 IC50 > 10000 nM T98698 C0LH8C 155511921 IC50 > 10000 nM T98698 CQ5BL7 155512551 IC50 > 50000 nM T98698 C5WUJ6 155513192 IC50 > 10000 nM T98698 CE4H7I 155513471 IC50 > 50000 nM T98698 CUKG21 155515602 IC50 > 50000 nM T98698 CA1J3N 155517086 IC50 = 6000 nM T98698 CL72ME 155517175 IC50 > 10000 nM T98698 CY54TU 155518062 IC50 = 100 nM T98698 CEH2N5 155518106 IC50 > 100000 nM T98698 CAD06U 155519254 IC50 = 500 nM T98698 CDY5H6 155519645 IC50 = 6400 nM T98698 CAZ3S7 155521187 IC50 = 15000 nM T98698 CZ75FW 155521272 IC50 = 8800 nM T98698 C49NGT 155529137 IC50 > 50000 nM T98698 CK2UY4 155531957 IC50 = 3200 nM T98698 CIZ46A 155533876 IC50 > 30000 nM T98698 C6LB5D 155535084 IC50 > 30000 nM T98698 C91UNV 155535585 IC50 > 10000 nM T98698 CTF98X 155537473 IC50 = 9400 nM T98698 CAG9P4 155537573 IC50 = 4500 nM T98698 CLD19W 155539311 IC50 > 10000 nM T98698 CU6V4Q 155539319 IC50 > 50000 nM T98698 C2UN1K 155545446 IC50 > 10000 nM T98698 C1JSY3 155545907 IC50 > 10000 nM T98698 CF2O4J 155546325 IC50 > 50000 nM T98698 CS3GO2 155546558 IC50 = 3200 nM T98698 C4Z5JX 155550827 IC50 > 50000 nM T98698 CH8L1V 155554197 IC50 > 10000 nM T98698 CGDF76 155554360 IC50 = 22000 nM T98698 CF2H3O 155555451 IC50 > 10000 nM T98698 CM7FN8 155555499 IC50 > 10000 nM T98698 CH0Z1P 155561539 IC50 > 10000 nM T98698 CGL24S 155562249 IC50 = 6200 nM T98698 CPNA06 155564750 IC50 > 50000 nM T98698 CD05RS 155566122 IC50 = 10000 nM T98698 C4A0RK 155566461 IC50 > 50000 nM T98698 C04CGS 155567444 IC50 = 15000 nM T98698 CS03PJ 155568350 IC50 > 50000 nM T98698 D00KFF 9882812 Ki = 4.7 nM T98698 D01YBR 44591988 IC50 = 33700 nM T98698 D02NWS 279980 IC50 = 150000 nM T98698 D03BQS 45482666 IC50 = 260 nM T98698 D03QOD 239512 IC50 = 650 nM T98698 D04KQF 6675804 Ki = 5426.9 nM T98698 D04UVL 1133083 IC50 > 50000 nM T98698 D05OVV 11993691 IC50 = 530 nM T98698 D06IMY 44626296 IC50 = 50 nM T98698 D09RKA 72946782 IC50 = 5000 nM T98698 D0A4HF 45482630 IC50 = 440 nM T98698 D0E0TA 44454650 IC50 > 50000 nM T98698 D0E9DD 16095101 IC50 = 9700 nM T98698 D0FN5D 45482672 IC50 = 1760 nM T98698 D0I4RK 45482660 IC50 = 4800 nM T98698 D0K7QR 45269423 IC50 = 220 nM T98698 D0M9LJ 44454415 IC50 > 50000 nM T98698 D0MD7H 44454143 IC50 > 50000 nM T98698 D0N9AK 44138031 IC50 = 20000 nM T98698 D0PK9V 45482643 IC50 = 1400 nM T98698 D0Q2GM 44454416 IC50 > 50000 nM T98698 D0Q5DI 71462653 IC50 = 4460 nM T98698 D0Q5MC 24753719 IC50 = 10 nM T98698 D0R7JA 53344908 IC50 = 40 nM T98698 D0T0SK 44138032 IC50 = 2300 nM T98698 D0T4JQ 264 IC50 > 2000000 nM T98698 D0U8FC 759408 IC50 > 50000 nM T98698 D0Z8PX 24757913 IC50 > 10000 nM T62841 D0I6LH 107985 IC50 = 14 nM T62841 D05VXK 56848369 IC50 = 77000 nM T62841 D0CM5P 6737869 IC50 = 34000 nM T62841 D0Z4SW 56848967 IC50 = 243000 nM T62841 CZQF03 9589606 EC50 = 199.53 nM T62841 CH0JQ4 9696680 EC50 = 6309.57 nM T62841 CJ79ZS 9831050 EC50 = 4200 nM T62841 C8TRG1 9950925 IC50 = 5000000 nM T62841 CNY07E 10149969 IC50 = 67800 nM T62841 CI16WO 10232703 EC50 = 28183.83 nM T62841 C2BTQ1 10395438 EC50 = 25.12 nM T62841 CC41EQ 10483914 EC50 = 3000 nM T62841 CP1N9D 11557006 Ki = 600 nM T62841 CTO42L 25108278 EC50 = 30 nM T62841 CZO38G 25108279 EC50 = 7943.28 nM T62841 CJY10U 25108280 EC50 = 10000 nM T62841 CYN0U4 25108338 EC50 = 2511.89 nM T62841 CH27QL 25108339 EC50 = 125.89 nM T62841 CMWE08 25108340 EC50 = 25.12 nM T62841 C83RMZ 25108341 EC50 = 6309.57 nM T62841 CL6K2Z 25108342 EC50 = 50.12 nM T62841 C29JGO 44433860 EC50 = 700 nM T62841 CX1VT3 44433864 EC50 = 1000 nM T62841 CC19MI 44433865 EC50 = 1800 nM T62841 CK4U1Y 44433867 EC50 = 1900 nM T62841 C7O2NA 44433868 EC50 = 1100 nM T62841 CNI8S7 44433869 EC50 = 400 nM T62841 CC2X4D 44433871 EC50 = 900 nM T62841 CS6J3Z 44433872 EC50 = 500 nM T62841 CYTF75 44433873 EC50 = 600 nM T62841 CUB3R9 44433874 EC50 = 600 nM T62841 CASU09 44433875 EC50 = 2500 nM T62841 C2F4XC 44433877 EC50 = 1300 nM T62841 CPR27Y 44433878 EC50 = 5000 nM T62841 CI5CM4 44433880 EC50 = 3000 nM T62841 CZYW46 44433883 EC50 = 2800 nM T62841 CF90JN 44433885 EC50 = 1400 nM T62841 C9YA2Q 44433886 EC50 = 300 nM T62841 CKH5P3 44433887 EC50 = 1300 nM T62841 CQTL72 44433892 EC50 = 3300 nM T62841 C39BRL 44433894 EC50 = 1700 nM T62841 C7DCM0 44433900 EC50 = 300 nM T62841 C6T2VJ 44433902 EC50 = 160 nM T62841 CWX82D 44433903 EC50 = 100 nM T62841 C8W3KA 44433904 EC50 = 100 nM T62841 C67QDB 44433905 EC50 = 100 nM T62841 C0AW2I 44433906 EC50 = 590 nM T62841 C2Z5HR 44433907 EC50 = 14900 nM T62841 C78DSJ 44433908 EC50 = 15800 nM T62841 CNIS69 44433909 EC50 = 4800 nM T62841 C4FJ3Y 44433910 EC50 = 10300 nM T62841 CJA36H 44433911 EC50 = 800 nM T62841 COT1X0 44433912 EC50 = 100 nM T62841 CW3N9A 44433913 EC50 = 100 nM T62841 CVTD69 44433914 EC50 = 100 nM T62841 CNP5D4 44433915 EC50 = 1600 nM T62841 C8F2YR 44433916 EC50 = 100 nM T62841 CJ0H1W 44433917 EC50 = 100 nM T62841 CF6NY1 44433918 EC50 = 4300 nM T62841 CT9RV0 44433940 EC50 = 200 nM T62841 C98REM 44433947 EC50 = 170 nM T62841 CC25TI 44433948 EC50 = 600 nM T62841 C3FK7I 44433949 EC50 = 320 nM T62841 CKXO16 44433963 EC50 = 1200 nM T62841 CFK1A0 44433964 EC50 = 1000 nM T62841 CCNA17 44433965 EC50 = 1100 nM T62841 CQ6Z4N 44433966 EC50 = 2000 nM T62841 C5VZ8G 44433967 EC50 = 600 nM T62841 C04RTO 44433968 EC50 = 1200 nM T62841 CCH60Z 44433970 EC50 = 1200 nM T62841 CGP93I 44433971 EC50 = 3600 nM T62841 C78NPU 49788150 EC50 > 50000 nM T62841 CH14XL 49788153 EC50 > 100000 nM T62841 CL5A8W 49788154 EC50 > 4000 nM T62841 CMC39J 49788155 EC50 > 100000 nM T62841 CGV0Q5 49788311 EC50 = 199.53 nM T62841 C3VNW4 49788378 EC50 = 12589.25 nM T62841 CBL79Q 49788379 EC50 > 50000 nM T62841 C9NM2I 49788380 EC50 = 316.23 nM T62841 CWXQ13 49788381 EC50 = 1000 nM T62841 CU5K0J 49788439 EC50 = 408 nM T62841 CA14BD 49788440 EC50 = 1995.26 nM T62841 C4Q3EK 49788441 EC50 = 7100 nM T62841 CY9X3A 49788504 EC50 = 12589.25 nM T62841 C02BPK 49788505 IC50 = 57000 nM T62841 CP4W7E 49788574 IC50 = 2000 nM T62841 C45UPM 51351273 EC50 = 142 nM T62841 CC5ES7 51351274 EC50 = 311 nM T62841 C4KPY5 51351408 EC50 = 3500 nM T62841 C8FCZ1 51351409 EC50 = 6590 nM T62841 C0P5FT 52948093 EC50 = 6100 nM T62841 C36PSZ 53318281 IC50 = 690 nM T62841 CUN9P6 53326692 EC50 = 138 nM T62841 CH4FR9 54582896 EC50 = 1400 nM T62841 CD86HV 56639666 IC50 = 400 nM T62841 C8UT1Y 56640042 EC50 = 1995.26 nM T62841 CLE0S5 56640398 IC50 = 8600 nM T62841 C2AW5B 56640474 IC50 = 1900 nM T62841 CY63EN 56640547 IC50 = 1200 nM T62841 C1U8GS 56640610 EC50 = 700 nM T62841 CDT76U 56640611 EC50 = 700 nM T62841 CESI03 57330164 IC50 = 1100 nM T62841 CNEO43 71511553 IC50 = 1258.93 nM T62841 CXB78U 73346321 EC50 = 200 nM T62841 CA41PT 73347818 IC50 = 700000 nM T62841 C7NTU0 73355411 EC50 = 4 nM T62841 CZO78P 117977940 IC50 = 4.8 nM T62841 CTH0N8 117978042 IC50 = 2 nM T62841 CSQ7N6 117990832 IC50 = 4400 nM T62841 CD21PQ 117991137 IC50 = 2 nM T62841 C0UDR9 126961334 IC50 = 4200 nM T62841 CW03MF 126961335 IC50 < 2.5 nM T62841 CO6M2S 127035718 Ki = 1940 nM T62841 C14WCD 127035910 Ki = 627 nM T62841 C8MOC4 127036298 IC50 = 2800 nM T62841 C3MTV5 127036301 IC50 > 10000 nM T62841 C8MC6H 134137699 IC50 = 8900 nM T62841 CY8N3X 134143255 IC50 = 3100 nM T62841 C9CS4G 134147747 EC50 = 700 nM T62841 C6BSE1 137633152 EC50 = 398.11 nM T62841 CS9UM8 137637330 EC50 = 199.53 nM T62841 CPXI31 137638214 EC50 = 95 nM T62841 C6W5BL 137641156 EC50 = 62 nM T62841 CJ8EN5 137643158 EC50 > 100000 nM T62841 CZ2W3S 137650859 EC50 > 100000 nM T62841 CD25WP 137653967 EC50 = 79.43 nM T62841 CW4D2N 137654325 EC50 = 31.62 nM T62841 C3V9ZC 137654661 EC50 = 79.43 nM T62841 C9F1TA 137661916 EC50 = 18 nM T62841 CA8EX2 145962815 IC50 = 6000 nM T62841 CPX6Q0 155512671 IC50 > 50000 nM T62841 C2ORE8 155534488 IC50 = 2 nM T62841 CQN9L7 155536026 IC50 > 50000 nM T62841 CFDM94 155549751 IC50 = 3300 nM T62841 CN4WT6 155564785 IC50 > 50000 nM T62841 CENS94 155567301 IC50 = 860 nM T62841 CYSM34 44433870 EC50 = 400 nM T56104 CN0FH2 2726759 IC50 = 3100 nM T56104 CL4XQ8 2826416 IC50 = 26600 nM T56104 CX6PS7 2826419 IC50 = 26600 nM T56104 CONM79 135473042 IC50 = 6300 nM T45758 CP37AU 16143282 IC50 = 9900 nM T45758 CJ94DY 16159336 IC50 = 78 nM T45758 CTD0I2 52946800 IC50 = 50 nM T55616 D0T9HG 132519 IC50 = 3.4 nM T55616 CSIB97 9896504 IC50 > 30000 nM T55616 C6MSI0 10141443 IC50 = 2000 nM T55616 CV5X8A 10224181 IC50 > 30000 nM T55616 C7XE1L 10437629 IC50 = 350 nM T55616 CR2UN0 11669859 IC50 = 5.7 nM T55616 CF75MS 23017979 IC50 = 3000 nM T55616 CQJ3S4 23018008 IC50 = 600 nM T55616 CVR52U 25066764 IC50 > 25 nM T55616 C3YAF6 44329898 IC50 = 550 nM T55616 C9R1ZE 44330132 IC50 = 4000 nM T55616 CLU8I7 44330135 IC50 = 220 nM T55616 C1IE0S 44330147 IC50 = 4000 nM T55616 CPG7N2 44330149 IC50 = 350 nM T55616 CYP6S4 44330152 IC50 = 1100 nM T55616 CMGA28 44330163 IC50 = 2500 nM T55616 CDO15M 118721026 IC50 = 24.7 nM T55616 CHO72Q 118721027 IC50 = 3260 nM T01973 D01PZD 5329098 IC50 > 10000 nM T01973 D03ZBT 11626560 IC50 = 300 nM T01973 D0G6QF 3081361 IC50 = 3370 nM T01973 D0IQ6P 25102847 IC50 = 69 nM T01973 D00DRL 44137946 IC50 = 7 nM T01973 D03LWG 53235510 IC50 = 2891 nM T01973 D05OMT 45142457 IC50 = 7 nM T01973 D06EGV 44603533 IC50 = 1.2 nM T01973 D07EHV 44814409 IC50 > 10000 nM T01973 D0D1GF 42642645 IC50 = 3 nM T01973 D0E3TC 44259 IC50 = 149 nM T01973 D0O6WV 24794418 IC50 = 1.8 nM T01973 D0T3ME 156422 IC50 > 30000 nM T01973 C6Y9CV 151193 IC50 > 10000 nM T01973 CUJR40 10062694 EC50 > 2000 nM T01973 CACS26 11561968 Ki > 2000 nM T01973 CU0E8O 11690457 Ki > 2000 nM T01973 CI7DT1 11857432 Ki = 581 nM T01973 CBT94Q 11857507 Ki = 79 nM T01973 CEA7I9 11857949 Ki = 80 nM T01973 CHR92S 11858109 Ki = 28 nM T01973 CDKH57 11858286 Ki = 706 nM T01973 CGC34R 16118737 IC50 > 25000 nM T01973 C2UV9Y 16222392 IC50 = 7 nM T01973 CA3I4T 24753787 IC50 > 50000 nM T01973 CQNP54 24764449 IC50 = 10 nM T01973 C4Z9CN 24769780 Ki = 1.3 nM T01973 CS0P4K 25054599 IC50 = 1030 nM T01973 C2F1YJ 25054600 IC50 = 410 nM T01973 C8CA3Y 25054857 IC50 = 60 nM T01973 CDYM40 25055101 IC50 = 12 nM T01973 CMH4W3 25055102 IC50 = 150 nM T01973 CQZ95L 25055103 IC50 = 590 nM T01973 C8UGB1 25055104 IC50 > 1000 nM T01973 CAE17C 25055344 IC50 > 1000 nM T01973 C4AR9G 25268137 IC50 = 60 nM T01973 CAK0F2 44155856 IC50 < 3 nM T01973 CNJ3Y1 44181654 IC50 = 25 nM T01973 CF6SL7 44256410 IC50 = 14 nM T01973 CYV2D7 44368815 IC50 > 10000 nM T01973 C3VRO9 44557921 IC50 > 10000 nM T01973 CD2CQ0 44564593 IC50 = 170 nM T01973 CYT37A 46232443 IC50 = 3600 nM T01973 C48ZVW 46232555 IC50 = 450 nM T01973 CS9B1U 46232556 IC50 = 230 nM T01973 CCXK70 46888806 IC50 = 200 nM T01973 C40DPT 46888807 IC50 = 80 nM T01973 CZB8P0 46888808 IC50 = 30 nM T01973 C7K9CZ 46888809 IC50 = 90 nM T01973 C0VSL7 46888810 IC50 = 100 nM T01973 CIXV03 46888811 IC50 = 30 nM T01973 C6UH7Y 46888812 IC50 = 40 nM T01973 C84SJR 46888813 IC50 = 90 nM T01973 CE1JL7 46889250 IC50 = 16 nM T01973 COT4E8 46889251 IC50 > 10000 nM T01973 CQ27HK 46889273 IC50 = 210 nM T01973 CS9G6E 50997096 IC50 > 10000 nM T01973 CEQN27 52936621 Ki > 1000 nM T01973 CM24LF 52938983 IC50 = 277.1 nM T01973 C09SDH 53257410 IC50 > 10000 nM T01973 CBK9Q6 53357848 IC50 = 50.4 nM T01973 C8NA4L 53384644 IC50 > 30000 nM T01973 C1XS2J 54760383 IC50 > 10000 nM T01973 CY3V6S 54764326 IC50 > 10000 nM T01973 CM8JX1 56604907 Ki = 1 nM T01973 CPHX64 57325478 IC50 > 50000 nM T01973 CQ9BW4 57325479 IC50 > 50000 nM T01973 C59OYH 57398540 IC50 > 10000 nM T01973 CF94GH 57812483 IC50 = 130 nM T01973 CVK0G4 58056356 IC50 > 50000 nM T01973 C1MR8Q 60097495 IC50 > 1000 nM T01973 C9ZCT2 62705065 IC50 = 336.4 nM T01973 C10AMI 66553589 IC50 = 8260 nM T01973 CV63UL 67240318 IC50 > 10000 nM T01973 C1BCX0 71579696 IC50 = 446 nM T01973 CED8U9 71601485 IC50 = 861 nM T01973 CHA9O3 71601634 IC50 = 2293 nM T01973 CBSF14 71601639 IC50 = 912 nM T01973 C0VOJ8 71601790 IC50 = 403 nM T01973 C1FAU8 71679855 IC50 = 18.7 nM T01973 C60TUV 72737208 IC50 = 6097 nM T01973 CJ3WA6 72737404 IC50 > 10000 nM T01973 CVNW01 73386831 IC50 > 1000 nM T01973 CCJ43A 86302281 IC50 > 10000 nM T01973 CPG3A5 86302574 IC50 > 30000 nM T01973 CX29IY 90655145 IC50 > 10000 nM T01973 C8F7XO 92131166 IC50 = 345.7 nM T01973 CWO9B7 118715995 IC50 = 28.6 nM T01973 CGSI94 122179285 IC50 = 10 nM T01973 C2TF6E 122179286 IC50 = 13 nM T01973 CM04OW 122179287 IC50 = 17 nM T01973 C4YR9I 122179288 IC50 = 95 nM T01973 CJ76AF 122179289 IC50 = 44 nM T01973 C1T7CU 122179290 IC50 = 575 nM T01973 C08KEM 122179540 IC50 = 6100 nM T01973 CG0RP7 122179547 IC50 = 5000 nM T01973 C1A0SQ 122179548 IC50 = 4800 nM T01973 CWA94G 122182409 IC50 = 270 nM T01973 C53FOD 122186955 IC50 = 23 nM T01973 CGB2M4 122186956 IC50 = 32 nM T01973 C3DQG0 122186957 IC50 = 45 nM T01973 C2QP6A 122186958 IC50 = 101 nM T01973 CYA03Q 122186959 IC50 = 25 nM T01973 CHL1E7 122186961 IC50 = 23 nM T01973 CK48SW 122186962 IC50 = 27 nM T01973 C4GIB5 122186963 IC50 = 14 nM T01973 C1R8VS 122187846 IC50 = 49 nM T01973 C3X8BL 122187848 IC50 = 34 nM T01973 CPC26B 122187849 IC50 = 30 nM T01973 C8KXV1 127025843 IC50 > 1000 nM T01973 CKS28E 127034802 IC50 = 93.4 nM T01973 CUO0C5 132156633 IC50 > 10000 nM T01973 C53OJM 132607333 IC50 = 82.56 nM T01973 CERS64 132937256 IC50 > 30000 nM T01973 CUKE45 134147919 IC50 = 140.72 nM T01973 CYL5V1 134694986 IC50 = 731 nM T01973 CJ7U4C 136053657 IC50 = 14.5 nM T01973 C4G5IA 137125270 IC50 = 361 nM T01973 CE75QD 137321162 IC50 = 2.9 nM T01973 C7TG3J 137641313 IC50 > 19952.62 nM T01973 C4HB8M 145949394 IC50 = 3.1 nM T01973 C2MD1Q 155513187 IC50 > 10000 nM T01973 C7SF2C 155547229 IC50 = 375 nM T01973 C40IYS 155562258 IC50 = 346 nM T01973 D00TBD 10461815 IC50 = 68 nM T01973 D06HVH 54613583 IC50 > 10000 nM T01973 D07OXC 11650194 Ki = 195 nM T01973 D0EE6A 6398883 IC50 > 10000 nM T01973 D0Q0YV 24944925 IC50 > 19952.62 nM T01973 D0R2WK 16038120 IC50 = 1634 nM T89055 D04XVN 11707110 IC50 = 1.6 nM T89055 D0E3TC 44259 IC50 = 37.4 nM T89055 D0K0YC 9826528 IC50 = 110 nM T89055 D0A9KI 9863367 IC50 > 50 nM T89055 C8KED5 4713 IC50 = 50000 nM T89055 CQ7PL4 1235170 IC50 > 20000 nM T89055 C5VPH9 16129448 IC50 = 391 nM T89055 C0H8UN 16730109 IC50 > 30000 nM T89055 C6P1CX 25066843 IC50 > 20000 nM T89055 C3VRO9 44557921 IC50 > 10000 nM T89055 CIPX17 45485590 Ki = 9700 nM T89055 CI10RQ 45485600 Ki = 13000 nM T89055 CPVU61 45485609 Ki = 6200 nM T89055 C58VXQ 45485625 Ki = 710 nM T89055 CMI83V 45485640 Ki = 2400 nM T89055 CP87FU 45485645 Ki = 1400 nM T89055 CLJF04 45485646 Ki = 1800 nM T89055 CQE7Z0 45485654 Ki = 3700 nM T89055 C5J4CW 45485664 Ki = 1400 nM T89055 C63VLU 45485665 Ki = 1800 nM T89055 C7VRC1 45485666 Ki = 2100 nM T89055 CK8Q9R 45485676 Ki = 16000 nM T89055 C7SX0U 45485677 Ki = 670 nM T89055 C4UB6E 45485687 Ki = 1400 nM T89055 CRA74I 49842779 IC50 = 6840 nM T89055 C37NKO 67129970 IC50 > 10000 nM T89055 CK80LJ 67130050 IC50 > 10000 nM T89055 CV63UL 67240318 IC50 > 10000 nM T89055 C7GRV2 68755406 IC50 > 10000 nM T89055 C2LAM7 126591927 IC50 = 82 nM T89055 CI2YE9 132606873 IC50 = 186.7 nM T89055 C0TE5S 135651612 IC50 = 1300 nM T89055 CI1E8V 137634241 IC50 > 10000 nM T89055 CU62AO 145712394 IC50 = 590 nM T89055 C6VB3O 145925651 IC50 >= 5000 nM T89055 C2MD1Q 155513187 IC50 > 10000 nM T89055 C4NKP6 155518298 IC50 = 1500 nM T89055 C86HPW 155518524 IC50 = 74000 nM T89055 D08LYB 5166 IC50 > 50 nM T89055 D0GD8Y 3006531 IC50 = 58 nM T48703 D06CTE 57469 EC50 > 270000 nM T48703 D08JWC 46241268 EC50 = 9000 nM T48703 D0C8KF 159603 EC50 = 4000 nM T48703 CW9OJ4 130714 EC50 > 270000 nM T48703 CE5O7L 617291 IC50 = 290 nM T48703 C10PMR 2740876 IC50 = 1400 nM T48703 CEO4Y8 2741936 IC50 = 1640 nM T48703 CAB40T 2772288 EC50 = 7300 nM T48703 CTG57E 2990940 IC50 = 9200 nM T48703 CSBO32 4575362 IC50 = 20000 nM T48703 CT1Z0W 10198719 EC50 = 1320 nM T48703 CQ8M2D 15034539 EC50 = 3960 nM T48703 C0G8ZK 16042898 EC50 < 100000 nM T48703 C53LHI 16222788 EC50 < 100000 nM T48703 C0TM6X 21470208 EC50 = 100 nM T48703 C01JYU 23079483 EC50 > 10000 nM T48703 C7J6ID 43148784 EC50 = 3230 nM T48703 CG51KI 43661477 EC50 = 4570 nM T48703 CWX2U5 44821558 IC50 = 35500 nM T48703 CJD3L4 46173651 EC50 = 6700 nM T48703 C8OK9G 52944297 EC50 = 14 nM T48703 C3PU5J 52945312 EC50 = 55 nM T48703 C9CY4L 54760856 IC50 > 10000 nM T48703 CV2R1D 56954508 IC50 = 50 nM T48703 CMX4D3 56954509 IC50 = 15630 nM T48703 CNG97O 56954510 IC50 = 10920 nM T48703 CD63TK 56954511 IC50 = 4650 nM T48703 C7ZR3S 56954831 IC50 = 4780 nM T48703 CN1DX0 57139455 EC50 = 73200 nM T48703 C8J4TX 57279993 EC50 = 22000 nM T48703 CV72GW 67181623 EC50 = 131000 nM T48703 CK2V9S 67182494 EC50 = 57000 nM T48703 C8P9WA 67183000 EC50 = 29000 nM T48703 CMO74J 67185919 EC50 = 260000 nM T48703 CZ1DF2 67607124 EC50 = 1800 nM T48703 CDCT67 68322071 EC50 = 231000 nM T48703 C8QA9E 68417258 EC50 = 3700 nM T48703 C9JMR1 70676948 EC50 = 6930 nM T48703 C4M7EO 70676949 EC50 = 10580 nM T48703 CZ2SQ7 70676950 EC50 = 4910 nM T48703 C92UGS 70677104 EC50 = 9790 nM T48703 C7YN2I 70677106 EC50 = 1680 nM T48703 CW69JB 70677107 EC50 = 3370 nM T48703 CS2Y5P 70677263 EC50 = 9380 nM T48703 CHD4Z6 70677264 EC50 = 5810 nM T48703 C2CF5M 70677266 EC50 = 9010 nM T48703 C7BRX3 70677268 EC50 = 4990 nM T48703 C8R7IY 70677407 EC50 = 7640 nM T48703 CBM1N7 70677537 EC50 = 2250 nM T48703 CA87JR 70677538 EC50 = 370 nM T48703 C7VFG9 70677539 EC50 = 850 nM T48703 CR9AY7 71284052 EC50 = 20860 nM T48703 C54YUS 71292238 EC50 > 270000 nM T48703 C61EPX 71292267 EC50 = 1500 nM T48703 CXQ26G 71292269 EC50 = 2700 nM T48703 CS4AF1 71292276 EC50 = 4400 nM T48703 CR6QJ7 71292278 EC50 = 4900 nM T48703 CDN7K8 71462538 EC50 = 4270 nM T48703 CMR0W9 71505363 EC50 = 7200 nM T48703 CWB56Z 71505551 EC50 = 31000 nM T48703 C0ML8V 72771075 EC50 = 1600 nM T48703 CU6HD7 73294130 EC50 = 24400 nM T48703 C17WYQ 73294131 EC50 = 46200 nM T48703 C8YL9F 80068544 EC50 = 7210 nM T48703 CC9J0R 85770050 IC50 = 7260 nM T48703 CR2F9W 86302334 EC50 = 200 nM T48703 CQ5Z9B 90647157 EC50 = 1130 nM T48703 C2TQN1 113393023 EC50 = 3740 nM T48703 CCX61Z 115552153 EC50 = 6610 nM T48703 C21YTZ 117889806 EC50 = 6600 nM T48703 C1C7HK 117890334 EC50 = 5010 nM T48703 CYN9O7 117908192 EC50 = 7120 nM T48703 CN6U9R 117908193 EC50 = 1650 nM T48703 CC3KG7 118711984 EC50 = 3160 nM T48703 CBGA29 121231447 EC50 = 49 nM T48703 C16IGR 121231448 EC50 = 27 nM T48703 CA20ET 122192082 EC50 = 150 nM T48703 CGA45W 122192084 EC50 = 120 nM T48703 C6EM8V 122192086 EC50 = 190 nM T48703 C5Z8VB 122192088 EC50 = 250 nM T48703 C4W2YX 122192092 EC50 = 38 nM T48703 CTMB98 122192093 EC50 = 1000 nM T48703 CQ46DT 122192097 EC50 = 699 nM T48703 C62EAW 122192098 EC50 = 91 nM T48703 C1K0FH 122192099 EC50 = 9 nM T48703 CD0U6Q 122192100 EC50 = 56 nM T48703 C8GDS5 122192101 EC50 = 2181 nM T48703 CI6P2L 122192102 EC50 = 2862 nM T48703 C29KEI 122192103 EC50 = 727 nM T48703 CTXN14 122192104 EC50 = 519 nM T48703 C7VRF9 122192105 EC50 = 1016 nM T48703 C45QVS 122192106 EC50 = 60 nM T48703 C8JUX9 122192107 EC50 = 50 nM T48703 CIE72N 122192108 EC50 = 85 nM T48703 C3G7EJ 122192110 EC50 = 621 nM T48703 CXC4S0 130276131 EC50 = 49800 nM T48703 C5T0QR 130289621 EC50 = 26700 nM T48703 CWEM85 130289681 EC50 = 3850 nM T48703 CJH93E 130289687 EC50 = 5340 nM T48703 CJY9E3 130289827 EC50 = 2210 nM T48703 CFQ95P 130708144 EC50 = 8500 nM T48703 C45BQH 132585194 EC50 = 13450 nM T48703 CUV27F 134106001 EC50 = 1640 nM T48703 CWAF78 135260389 EC50 = 2350 nM T48703 C7WG8O 135260399 EC50 = 1310 nM T48703 C7EYM0 135260402 EC50 = 2700 nM T48703 C15GPU 135260404 EC50 = 3140 nM T48703 C0OC5M 135260416 EC50 = 1220 nM T48703 CEN0Y8 135260422 EC50 = 2310 nM T48703 CC8SJ4 135260424 EC50 = 453 nM T48703 C96OZB 135260428 EC50 = 1050 nM T48703 C02NFK 135271001 EC50 = 3280 nM T48703 CF1J7O 135271003 EC50 = 780 nM T48703 CBZ3L0 135271004 EC50 = 20000 nM T48703 CLK27F 135271006 EC50 = 1200 nM T48703 C2JXW8 135271007 EC50 = 1220 nM T48703 CGD0Y6 135271008 EC50 = 178 nM T48703 CQS26J 135271009 EC50 = 34000 nM T48703 COC2D9 135271011 EC50 = 1660 nM T48703 C6KGY3 135271012 EC50 = 126 nM T48703 CX15DN 135271013 EC50 = 3790 nM T48703 CRE58J 135271014 EC50 = 280 nM T48703 CF8AX4 135271016 EC50 = 366 nM T48703 C4LX5U 135271017 EC50 = 29 nM T48703 COL31X 135271018 EC50 = 203 nM T48703 CSK9J6 135271020 EC50 = 5000 nM T48703 CB8J0D 135271022 EC50 = 254 nM T48703 C30AKS 135271027 EC50 = 4900 nM T48703 CK5FB8 135271028 EC50 = 133 nM T48703 CWG6U8 135271030 EC50 = 1100 nM T48703 CB6J0X 135271031 EC50 = 1050 nM T48703 CTSI07 135271032 EC50 = 857 nM T48703 CWL20P 135271033 EC50 = 167 nM T48703 C29UTE 135271034 EC50 = 92 nM T48703 C9K2QF 135271035 EC50 = 300 nM T48703 C5N3YE 135271038 EC50 = 110 nM T48703 CB3G8N 135271039 EC50 = 128 nM T48703 CN6U7D 135271040 EC50 = 16200 nM T48703 CJDE91 135271042 EC50 = 830 nM T48703 CO7CT1 135271043 EC50 = 749 nM T48703 CC2S6G 135271044 EC50 = 1190 nM T48703 CE0F5R 135271045 EC50 = 179 nM T48703 C8UBG3 137515213 EC50 > 100000 nM T48703 C5Q6TS 137515380 EC50 > 100000 nM T48703 CNT8G1 137515383 EC50 > 100000 nM T48703 CVI1H4 137515466 EC50 > 100000 nM T48703 CKC32Q 137515546 EC50 > 100000 nM T48703 C6Q5YE 137515571 EC50 > 100000 nM T48703 CJ85ER 137515794 EC50 > 100000 nM T48703 CSU98Z 137515846 EC50 > 100000 nM T48703 C0M6SU 137515935 EC50 > 100000 nM T48703 C4TGP3 137516041 EC50 > 100000 nM T48703 CS15BK 137516054 EC50 > 100000 nM T48703 C0F5XW 137516341 EC50 > 100000 nM T48703 CSH86R 137657602 EC50 = 9240 nM T48703 C0O6SE 137658022 EC50 = 500 nM T48703 CWUB82 146037590 IC50 = 30 nM T48703 CT81ZB 154734323 IC50 = 1040 nM T48703 CV4RP7 154734324 IC50 = 300 nM T48703 C4H1OC 155461355 IC50 = 10120 nM T48703 CV18UD 155461357 IC50 > 20000 nM T48703 CTV73B 155461358 IC50 = 110 nM T48703 C0NQC8 155461361 IC50 > 20000 nM T48703 CAM36I 155461362 IC50 > 20000 nM T48703 CW85TP 155461363 IC50 = 4840 nM T48703 CMS2J0 155461364 IC50 = 390 nM T48703 CLV76O 155461366 IC50 = 210 nM T48703 C2DPY6 155461367 IC50 = 2810 nM T48703 C8U5YH 155461369 IC50 = 980 nM T48703 CBE24O 155461370 IC50 = 350 nM T48703 CNTD39 155461371 IC50 = 190 nM T48703 C4E2DP 155461372 IC50 = 600 nM T48703 CM4T7B 155461373 IC50 = 3860 nM T48703 CL7NJ5 155461374 IC50 = 290 nM T48703 C68AXI 155461375 IC50 > 20000 nM T48703 CH3F8D 155461377 IC50 = 1060 nM T48703 CUJ36Z 155461378 IC50 = 520 nM T48703 C0SXQ3 155461379 IC50 = 630 nM T48703 CY9MI7 155461380 IC50 = 1180 nM T48703 CF0IW5 155461381 IC50 = 2080 nM T48703 CX71SQ 155461382 IC50 = 1610 nM T48703 C0B5MV 155461383 IC50 = 800 nM T48703 CQ7A9H 155461384 IC50 > 20000 nM T48703 C1UCW6 155461385 IC50 = 390 nM T48703 CS0V3W 155461390 IC50 = 550 nM T48703 C3FO1T 155461391 IC50 = 590 nM T48703 C4HG5W 155510901 IC50 = 2410 nM T48703 CS59AL 155511147 IC50 > 50000 nM T48703 CO83UF 155512391 IC50 = 2520 nM T48703 C5ELT6 155512682 EC50 = 300 nM T48703 C4PT7D 155516384 IC50 = 5000 nM T48703 CBR24X 155516810 IC50 = 5290 nM T48703 CJ57AV 155524947 IC50 = 1110 nM T48703 C6T1WC 155525693 IC50 = 2870 nM T48703 C35WAO 155526329 IC50 > 50000 nM T48703 CC0H8N 155527771 IC50 = 2320 nM T48703 CWG5Q4 155529545 IC50 > 50000 nM T48703 C8U0PK 155531703 IC50 > 50000 nM T48703 CHJ82Q 155532543 IC50 = 770 nM T48703 C2KF8C 155534024 IC50 = 1590 nM T48703 CA38PW 155537840 IC50 > 50000 nM T48703 CUB76Z 155540600 IC50 = 2630 nM T48703 CX5Z6H 155541402 IC50 = 2040 nM T48703 CT6F5Y 155543587 EC50 = 300 nM T48703 CXF3R7 155551884 IC50 = 3200 nM T48703 C13RUF 155552444 IC50 = 4020 nM T48703 CQ58RF 155556337 IC50 = 9000 nM T48703 CT79FB 155556399 IC50 = 6000 nM T48703 CB98NZ 155563615 IC50 = 3000 nM T48703 CV5R0M 155569666 IC50 = 880 nM T40243 CACS26 11561968 Ki > 10000 nM T40243 CU0E8O 11690457 Ki > 10000 nM T40243 CB0AP2 11705863 Ki > 10000 nM T40243 CEQN27 52936621 Ki > 1000 nM T40243 C1MR8Q 60097495 IC50 > 10000 nM T75797 D06FEA 5280360 EC50 = 250 nM T75797 D0WL5V 9867642 Ki = 9991 nM T75797 D00HTY 5280363 IC50 = 2.5 nM T75797 D00IQH 11677589 Ki > 5000 nM T75797 D00MZK 9911469 Ki > 10000 nM T75797 D08QWQ 5283081 EC50 = 12 nM T75797 D0K1EG 11508736 IC50 > 10000 nM T75797 CAZT67 1283333 IC50 = 4168.69 nM T75797 CLM8P6 2114670 Ki > 25000 nM T75797 CI4F0K 5282380 EC50 = 34.4 nM T75797 CK16QC 5311234 IC50 = 2 nM T75797 CO7N1Z 5311239 IC50 = 350 nM T75797 C4LY3F 6438324 EC50 = 2.7 nM T75797 CZ15QS 6441607 IC50 = 16 nM T75797 CC9BE3 6443852 EC50 = 4.1 nM T75797 C6TA3N 9809136 Ki = 5000 nM T75797 CV24TI 9817292 Ki > 83000 nM T75797 CYNX09 9825293 IC50 = 10 nM T75797 CKMW12 9874010 Ki = 6200 nM T75797 CF0HC5 9888589 IC50 = 42 nM T75797 CFC8G4 9894720 Ki > 3000 nM T75797 CA5N0K 9895436 Ki = 1300 nM T75797 CQ0X9R 9909510 IC50 = 76 nM T75797 CICE70 9938626 Ki = 5300 nM T75797 CWDT69 9939791 Ki = 3800 nM T75797 C6SGH7 9954562 Ki > 500 nM T75797 C4UK2Q 9955802 Ki > 3000 nM T75797 CZUJ52 10001608 IC50 = 42 nM T75797 CQ3GW6 10047541 IC50 = 11 nM T75797 CNE21V 10095268 IC50 < 3162.28 nM T75797 CEM21G 10181606 Ki = 17000 nM T75797 C0ED9Y 10251023 IC50 = 3 nM T75797 CL7YG3 10287121 Ki > 13000 nM T75797 C51JIX 10389527 EC50 = 85 nM T75797 CB19MW 10402929 Ki = 41000 nM T75797 C7G6QN 10551015 Ki = 1900 nM T75797 CI5HA0 10648334 IC50 = 320 nM T75797 C9YQG5 10670992 IC50 = 17 nM T75797 CC4OA3 10717894 Ki = 56000 nM T75797 C7GY6X 10739351 IC50 = 90 nM T75797 CY8IB2 10740699 IC50 = 1424 nM T75797 C12SBH 10741017 IC50 = 63 nM T75797 CG17HE 10741197 IC50 = 29 nM T75797 C87SIQ 10981979 IC50 = 311 nM T75797 CKST02 11122314 IC50 = 114 nM T75797 C1R0JI 11133176 IC50 = 4100 nM T75797 C0Y1TD 11133782 IC50 = 6700 nM T75797 C4S5MX 11249458 Ki > 10000 nM T75797 C70ESM 11269563 Ki > 20000 nM T75797 C9E4SW 11294166 Ki > 20000 nM T75797 CN2TG7 11387144 Ki > 1000 nM T75797 CXPO04 11408533 Ki > 20000 nM T75797 CZ4K0P 11476788 Ki = 21057 nM T75797 CE2JA4 11488860 Ki = 4320 nM T75797 C1W2ZK 11577792 Ki > 6000 nM T75797 C7Y6XJ 11597294 Ki = 14000 nM T75797 C51UDK 11667741 IC50 > 10000 nM T75797 C3BSV4 11696697 Ki > 13000 nM T75797 CNYK74 11743212 Ki = 22000 nM T75797 C93FZV 13174090 EC50 = 16 nM T75797 CT34LO 13230981 Ki > 13000 nM T75797 CO19GA 14372497 Ki > 20000 nM T75797 CB1N7G 14429703 EC50 = 1800 nM T75797 C06OGJ 15486805 IC50 = 12 nM T75797 C0L3VU 15486806 IC50 = 570 nM T75797 CWQ8B9 15551228 Ki > 500 nM T75797 CIS83K 15947857 Ki = 340 nM T75797 C3L0RK 15948325 Ki = 2000 nM T75797 CI61TE 16678098 IC50 > 10000 nM T75797 CX08BC 21198692 Ki > 500 nM T75797 CF81SW 23582412 IC50 > 10000 nM T75797 CP2S4J 23663736 Ki > 10000 nM T75797 C9H4WT 23686961 IC50 > 10000 nM T75797 CASU54 23696973 IC50 > 10000 nM T75797 C42LYP 24765153 Ki = 25700 nM T75797 CF72YI 24765671 Ki >= 785 nM T75797 C31JZP 24765672 Ki >= 2500 nM T75797 C4QX7Y 24765675 Ki >= 930 nM T75797 CL7Z9U 24765768 Ki >= 110 nM T75797 CFQA40 24952577 Ki > 7282 nM T75797 CD98IN 24952580 Ki > 456 nM T75797 C81WVN 24952927 Ki > 5474 nM T75797 CZT83E 24952928 Ki > 501 nM T75797 C8YHX3 24953283 Ki > 224 nM T75797 CZ93FO 24953285 Ki > 628 nM T75797 C17JTY 24953286 Ki > 2226 nM T75797 CFT0W5 24953624 Ki > 4992 nM T75797 C42VMD 24953625 Ki > 3461 nM T75797 C7B2EW 24953628 Ki > 2117 nM T75797 CXQJ67 25002382 Ki >= 1291 nM T75797 CN5SH9 25003075 Ki = 6400 nM T75797 C4J2BS 25195248 IC50 = 3800 nM T75797 CNOF71 44138108 Ki > 25700 nM T75797 CSRV98 44157014 IC50 = 3590 nM T75797 C2AV1K 44190762 IC50 = 2730 nM T75797 CR68BA 44250281 Ki > 25118.86 nM T75797 CN90FE 44269464 Ki > 13000 nM T75797 C1L0ET 44269468 Ki > 13000 nM T75797 C5KRQ4 44269486 Ki > 13000 nM T75797 CL6M2P 44269516 Ki > 13000 nM T75797 CON8R9 44269520 Ki > 13000 nM T75797 C6MBG0 44269521 Ki > 13000 nM T75797 CZ3Q1L 44269523 Ki > 13000 nM T75797 CRL61O 44269532 Ki > 13000 nM T75797 C1Z4LU 44269540 Ki > 13000 nM T75797 CM72FA 44269542 Ki > 13000 nM T75797 CN0JV2 44269543 Ki > 13000 nM T75797 C28UJH 44269544 Ki > 13000 nM T75797 CR1IY6 44269568 Ki > 13000 nM T75797 CI3C9O 44269596 Ki > 13000 nM T75797 CC0EW9 44269597 Ki > 13000 nM T75797 C9THI4 44285145 IC50 = 4400 nM T75797 CWJC89 44285146 IC50 = 630 nM T75797 CJ7DF5 44285161 IC50 = 3630 nM T75797 CBU0L2 44285199 IC50 = 2140 nM T75797 C5P9CF 44285208 IC50 = 210 nM T75797 CCD2S1 44285209 IC50 = 540 nM T75797 C9U7YH 44285251 IC50 = 290 nM T75797 C6EZ1R 44285252 IC50 = 1620 nM T75797 C5NV1S 44285270 IC50 = 5890 nM T75797 CS64GQ 44285310 EC50 > 20000 nM T75797 CDP9F2 44285328 IC50 = 210 nM T75797 CEYH21 44322291 IC50 = 350 nM T75797 CEGT75 44322535 IC50 = 11000 nM T75797 CS5UJ3 44322588 IC50 = 6100 nM T75797 C7VP5E 44322611 IC50 = 330 nM T75797 CW6H1J 44322613 IC50 = 32 nM T75797 C1C5VX 44354547 IC50 = 1000 nM T75797 CVC8B5 44354580 IC50 > 10000 nM T75797 CLN63A 44377464 Ki = 63000 nM T75797 C4F9NG 44393420 EC50 = 57 nM T75797 CD7JX6 44393422 EC50 = 252 nM T75797 CY26OC 44393431 EC50 = 67 nM T75797 C04DYE 44393436 EC50 = 58 nM T75797 CP71XZ 44393438 EC50 = 194 nM T75797 CE8G7U 44393443 EC50 = 899 nM T75797 CS78NL 44393448 EC50 = 23 nM T75797 CY0Z3L 44393451 EC50 = 249 nM T75797 C9OZ0V 44393457 EC50 = 781 nM T75797 C1M3TO 44393462 EC50 = 187 nM T75797 CL2FP6 44393474 EC50 = 2380 nM T75797 C8B6TD 44393475 EC50 > 10000 nM T75797 C6T2US 44393601 EC50 = 293 nM T75797 C78ANV 44393607 EC50 = 573 nM T75797 CWL1X4 44400355 Ki > 1000 nM T75797 CIB2W5 44419347 Ki > 500 nM T75797 C91JXT 44419374 Ki > 500 nM T75797 CNF4W2 44419379 Ki > 500 nM T75797 CDBE16 44450497 Ki > 24826 nM T75797 CUHD74 44564571 IC50 = 2400 nM T75797 CA05LN 44564804 IC50 = 1970 nM T75797 C6XE0K 44564841 IC50 = 3190 nM T75797 CND54C 44564892 IC50 = 4640 nM T75797 C2VR6S 44564893 IC50 = 3570 nM T75797 C18GXI 44564937 IC50 = 3160 nM T75797 CZ74GB 44564990 IC50 = 2230 nM T75797 C0NF1S 44565193 IC50 = 1820 nM T75797 CJKA53 44570666 IC50 = 16400 nM T75797 CSW92V 44570668 IC50 = 7400 nM T75797 CTW6L7 44570712 IC50 = 7600 nM T75797 CGX17U 44571206 IC50 = 10200 nM T75797 C5URT2 44571290 IC50 = 27400 nM T75797 CE4UO5 44571291 IC50 = 6100 nM T75797 CK1GW9 44571352 IC50 = 4200 nM T75797 CXQI89 44571354 IC50 = 6400 nM T75797 CS4F0X 46879894 IC50 = 600 nM T75797 C2FR7X 46885690 IC50 > 20000 nM T75797 CN8D5V 46885691 IC50 > 20000 nM T75797 C9RP0X 46885735 IC50 > 20000 nM T75797 C0A2CI 46890616 Ki >= 504 nM T75797 CW52VH 46890658 Ki >= 260 nM T75797 CXQ2W0 46890659 Ki >= 580 nM T75797 CQ20RC 46890660 Ki >= 100 nM T75797 CTR7Q0 49850345 IC50 > 50118.72 nM T75797 CM06FG 50898361 Ki > 8700 nM T75797 C4K6BH 52946883 Ki > 10000 nM T75797 CWR1Z7 56665984 Ki > 13000 nM T75797 CI0A9L 68747456 EC50 = 530 nM T75797 C6IHR3 68747472 EC50 = 640 nM T75797 C5NZO0 68747479 EC50 = 28 nM T75797 C8MED0 68749474 EC50 = 22 nM T75797 CIUR89 68751402 EC50 = 73 nM T75797 C8WC4E 68785185 EC50 = 3.8 nM T75797 CJ7AY6 69753740 EC50 = 7.1 nM T75797 C5WR8L 71450954 IC50 = 71 nM T75797 CSJ4A9 118352160 EC50 > 10000 nM T75797 CE6L8I 118352177 EC50 > 10000 nM T75797 C8PKA7 118352211 EC50 > 10000 nM T75797 CPS7M4 118352285 EC50 > 10000 nM T75797 C8ZRJ0 126495398 EC50 > 10000 nM T75797 C8SRZ5 126495427 EC50 > 10000 nM T75797 CD72CT 126495432 EC50 > 10000 nM T75797 CN72WL 126495463 EC50 > 10000 nM T75797 CV1A6C 126495491 EC50 = 8500 nM T75797 CYP3E5 126495507 EC50 > 10000 nM T75797 CX9M6D 127029402 EC50 > 10000 nM T75797 CWXR72 127029417 Ki > 50000 nM T75797 CW1O4F 127029692 EC50 > 10000 nM T75797 CJAQ90 127047381 Ki > 50000 nM T75797 CTR62O 127052613 EC50 = 32 nM T75797 CGZR45 127052614 EC50 = 380 nM T75797 COVY75 127052615 EC50 > 10000 nM T75797 C4U3XA 134138103 EC50 = 43 nM T75797 C10OQL 134144861 EC50 = 880 nM T75797 CG0SO1 134147356 EC50 = 280 nM T75797 C8QT5L 134149776 EC50 = 110 nM T75797 C16HYX 134151657 EC50 = 110 nM T75797 CIA76T 134157766 EC50 = 1000 nM T75797 D02MXT 24952929 Ki > 24000 nM T75797 D03OYD 5311240 IC50 = 1 nM T75797 D05TNX 5311100 EC50 = 3.6 nM T75797 D07UDT 15551229 Ki > 500 nM T75797 D0O9ES 5311053 IC50 = 1 nM T75797 D0S2LO 9864831 Ki > 13000 nM T75797 D0TA0L 23685469 Ki > 1000 nM T75797 D0Y1IF 23664784 Ki > 1000 nM T75797 D0Z3XJ 9817405 Ki > 500 nM T37154 D00UVA 11556711 IC50 > 30000 nM T37154 D0B2OT 5936 IC50 = 10000 nM T37154 D0SH3I 387447 IC50 = 9200 nM T37154 C1F3PN 53308743 IC50 = 26 nM T37154 C8U4OD 56649692 IC50 = 1000000 nM T37154 C7UTZ3 60182323 IC50 = 5 nM T37154 C7ZCG5 67362057 IC50 = 10 nM T37154 CC5B4K 67362073 IC50 = 3 nM T37154 C5MV0X 67362514 IC50 = 70 nM T37154 C80FME 67362517 IC50 = 50 nM T37154 CR46HB 71449876 IC50 = 15 nM T37154 CHI16O 71449892 IC50 = 87 nM T37154 C8KC7R 71449893 IC50 = 200 nM T37154 CDUY41 71451691 IC50 = 70 nM T37154 CP2W3G 71451692 IC50 = 59 nM T37154 C8OKN2 71451708 IC50 = 102 nM T37154 CFHD61 71451709 IC50 = 226 nM T37154 C31HBO 71453540 IC50 = 120 nM T37154 CJ6T7O 71455231 IC50 = 15 nM T37154 C0TGA7 71455232 IC50 = 100 nM T37154 CD4KH3 71457028 IC50 = 7800 nM T37154 CUJK72 71458886 IC50 = 375 nM T37154 CGC0P4 71458887 IC50 = 110 nM T37154 CR5K9Y 71458888 IC50 = 110 nM T37154 C7PDN8 71460698 IC50 = 5380 nM T37154 C4JK9N 71460699 IC50 > 30000 nM T37154 CO4E9Y 71460700 IC50 = 30 nM T37154 CF9MR5 71460701 IC50 = 76 nM T37154 CTG34V 71460713 IC50 = 252 nM T37154 CC6SX4 71462409 IC50 = 274 nM T37154 CC53AL 71462410 IC50 = 357 nM T37154 C5R2DM 71462411 IC50 = 803 nM T37154 CT1FB6 71462412 IC50 = 60 nM T37154 CU8PD3 71462413 IC50 = 100 nM T37154 CTAX32 71462414 IC50 = 25 nM T37154 C6A4BL 71462415 IC50 = 57 nM T37154 CFPT98 90655054 IC50 > 30000 nM T37154 C5JZ8R 90655055 IC50 > 30000 nM T37154 D09FGQ 123985 IC50 > 300000 nM T37154 D0F3CA 1609 IC50 = 600 nM T37154 D0I9PF 60182322 IC50 = 38 nM T83145 D0SH3I 387447 IC50 = 9.7 nM T83145 D0T3NB 5154 IC50 = 2000 nM T83145 D0U3EP 445154 IC50 = 2500 nM T83145 D0W0VD 3885 IC50 = 4000 nM T83145 D0Y2SW 25183872 IC50 = 6.2 nM T83145 D01OLO 9820526 IC50 = 8 nM T83145 C63WLY 89644 IC50 = 800 nM T83145 CC8QV4 124072 IC50 > 50000 nM T83145 CN0XJ3 439647 IC50 = 3800 nM T83145 CZ0AH3 638278 IC50 = 32000 nM T83145 CN71BS 641819 IC50 = 29000 nM T83145 C1KTS2 1371588 IC50 = 34000 nM T83145 C80RBM 3084606 IC50 = 11000 nM T83145 CA6Q2L 5282361 IC50 = 24000 nM T83145 CT0E7G 6293081 IC50 = 8000 nM T83145 C4A0NL 6436598 IC50 = 1060 nM T83145 C4ISO7 6438092 IC50 = 38000 nM T83145 CGW57O 6440856 IC50 = 7000 nM T83145 CPQ93K 9799505 IC50 = 14100 nM T83145 C4VG9X 9863590 IC50 = 20 nM T83145 C2TS1U 9907182 IC50 = 3 nM T83145 C6DBO0 9910975 IC50 = 50 nM T83145 CLWO04 10065309 IC50 = 200 nM T83145 C64YXB 10067871 IC50 = 45 nM T83145 CY69JC 10222612 IC50 = 25000 nM T83145 CUE3O7 10245314 IC50 = 35 nM T83145 CDK0O9 10316054 IC50 = 3400 nM T83145 C10MCP 10407641 IC50 = 50 nM T83145 CD0M8B 10499355 IC50 = 4000 nM T83145 CN0MX6 10525196 IC50 > 10000 nM T83145 C48SVD 10552343 IC50 > 10000 nM T83145 CKC1V4 10574522 IC50 > 10000 nM T83145 C9EUI1 10574991 IC50 = 10000 nM T83145 CN9S4F 10622840 IC50 > 10000 nM T83145 CT0QH3 10624842 IC50 = 800 nM T83145 CQ8W9A 10666813 IC50 = 300 nM T83145 C2GY5Z 10666814 IC50 = 1700 nM T83145 CJ16AD 10716177 IC50 > 10000 nM T83145 CJ5NW8 10716536 IC50 > 10000 nM T83145 C6C0JV 10716588 IC50 = 500 nM T83145 COE42S 10717756 IC50 > 30000 nM T83145 CNT0E3 10740841 IC50 = 400 nM T83145 C3XI4G 10741644 IC50 > 10000 nM T83145 C61PDW 10741998 IC50 = 400 nM T83145 C0VK9R 10759713 IC50 = 9400 nM T83145 C7K2EB 10763720 IC50 = 600 nM T83145 CON93J 10764421 IC50 > 10000 nM T83145 CB40RO 10786213 IC50 > 10000 nM T83145 C7BAM8 10787015 IC50 = 400 nM T83145 CGRH71 10811870 IC50 > 10000 nM T83145 C3GRB1 10813496 IC50 = 9800 nM T83145 CDAG94 11426529 IC50 = 37200 nM T83145 CW04NP 11842418 IC50 = 5500 nM T83145 CX2SH5 14632858 EC50 = 26070 nM T83145 CWFY96 15143722 IC50 > 10000 nM T83145 C4DU0A 15560077 IC50 = 1560 nM T83145 CK7JE6 16752764 IC50 = 10000 nM T83145 CHQ84E 21589810 IC50 = 5000 nM T83145 C0P5WS 24971029 IC50 > 10000 nM T83145 C6O4MS 25017848 IC50 = 1200 nM T83145 CMAH54 25017849 IC50 = 200 nM T83145 CSYN01 42631933 IC50 = 5500 nM T83145 CX3AJ7 42632173 IC50 = 1200 nM T83145 CKD03R 44241655 IC50 = 100 nM T83145 CV6F7Y 44289452 IC50 = 700 nM T83145 C5FP0H 44289467 IC50 = 5000 nM T83145 C2SW4U 44289470 IC50 = 900 nM T83145 CA8DQ9 44289488 IC50 = 1000 nM T83145 CDWJ01 44289501 IC50 = 700 nM T83145 C3MW8A 44289516 IC50 = 4000 nM T83145 C8ZNQ2 44289549 IC50 = 300 nM T83145 C6VG4T 44289672 IC50 = 10000 nM T83145 CN6P5R 44289703 IC50 = 6000 nM T83145 CQ4N8X 44289710 IC50 = 2000 nM T83145 CO6YJ1 44289723 IC50 = 1000 nM T83145 CH70YI 44289728 IC50 = 8000 nM T83145 C90ILK 44289729 IC50 = 6000 nM T83145 CTD61E 44289731 IC50 = 2000 nM T83145 CP61ET 44289744 IC50 = 300 nM T83145 CNX83C 44289751 IC50 = 200 nM T83145 CKC60H 44289752 IC50 = 5000 nM T83145 CB1U7R 44289768 IC50 = 7000 nM T83145 C41UCE 44289771 IC50 = 700 nM T83145 C43FXZ 44289772 IC50 = 200 nM T83145 CQS67E 44289780 IC50 = 200 nM T83145 CK05AX 44289781 IC50 = 100 nM T83145 CCF9N8 44289806 IC50 = 300 nM T83145 C8HQ1I 44289817 IC50 = 10000 nM T83145 C2LG7F 44289821 IC50 = 200 nM T83145 CRA6S8 44289830 IC50 = 20000 nM T83145 CK03UA 44289831 IC50 = 10000 nM T83145 C2UP0B 44289832 IC50 = 300 nM T83145 CPD2N6 44289849 IC50 = 15000 nM T83145 C7DMF0 44289850 IC50 = 7000 nM T83145 CZ24YP 44289858 IC50 = 10000 nM T83145 CD3XS5 44289873 IC50 = 3000 nM T83145 C7YLF3 44289889 IC50 = 1000 nM T83145 C51LTY 44289904 IC50 = 300 nM T83145 CKZ05A 44289907 IC50 = 200 nM T83145 C1S2LK 44289913 IC50 = 400 nM T83145 CLMF82 44289916 IC50 = 16000 nM T83145 CS74XH 44289917 IC50 = 10000 nM T83145 C01YUD 44290015 IC50 = 1000 nM T83145 CCA93I 44290016 IC50 = 4000 nM T83145 CD76MS 44290017 IC50 = 10000 nM T83145 C5LKN8 44290028 IC50 = 2000 nM T83145 CRA5C3 44290086 IC50 = 1000 nM T83145 C5T9MD 44320262 IC50 = 400 nM T83145 CA78EB 44320323 IC50 = 300 nM T83145 CP3RW2 44320513 IC50 = 98 nM T83145 C3G4YN 44320524 IC50 = 2000 nM T83145 CRWI45 44320559 IC50 = 210 nM T83145 CO3P4J 44320570 IC50 = 4400 nM T83145 CTF3J9 44346502 IC50 = 13500 nM T83145 CKEL64 44346503 IC50 = 11700 nM T83145 CI90EK 44346510 IC50 = 11700 nM T83145 C96XLU 44346547 IC50 = 13800 nM T83145 CU9JX1 44346548 IC50 = 28400 nM T83145 CR45YK 44346614 IC50 = 21300 nM T83145 CLF62A 44346695 IC50 > 50000 nM T83145 CGX1I9 44346696 IC50 > 50000 nM T83145 C7G4SQ 44346698 IC50 > 50000 nM T83145 CK54LZ 44346699 IC50 = 17500 nM T83145 CW32JB 44346700 IC50 = 17700 nM T83145 C3OD0W 44346701 IC50 > 50000 nM T83145 CTQO74 44346819 IC50 = 25500 nM T83145 C1GC4T 44346831 IC50 > 50000 nM T83145 CC9IR0 44346850 IC50 = 14100 nM T83145 CD38OI 44346867 IC50 > 50000 nM T83145 CUVQ80 44346868 IC50 > 50000 nM T83145 C8P2NF 44346888 IC50 = 16200 nM T83145 C87TYU 44346898 IC50 = 14100 nM T83145 C63MGJ 44346900 IC50 > 50000 nM T83145 CZ43OU 44346912 IC50 = 11800 nM T83145 CYC9O0 44560837 IC50 = 6420 nM T83145 C2ZXP8 45270718 IC50 = 30 nM T83145 CM81GQ 46864294 IC50 = 9 nM T83145 CWDL81 52948098 IC50 = 45 nM T83145 CXE1S6 56834952 IC50 = 9200 nM T83145 CG2D5M 57149553 IC50 = 900 nM T83145 C9SMV3 68815772 IC50 = 28300 nM T83145 C7R5EZ 71571581 IC50 > 50000 nM T83145 CVC61J 71699285 IC50 = 1020 nM T83145 C6Z8PV 71725229 IC50 = 33400 nM T83145 C43EHW 73346049 IC50 = 980 nM T83145 C5XO2M 73348950 IC50 > 50000 nM T83145 C7INR4 73356550 IC50 = 32300 nM T83145 CD65OQ 73356552 IC50 = 4600 nM T83145 CRK58L 84922307 IC50 = 23000 nM T83145 CJ3KU9 86294767 IC50 = 5000 nM T83145 CI4SU3 86294768 IC50 = 5800 nM T83145 C1LNM5 86294769 IC50 = 2400 nM T83145 CJ0T6L 86294770 IC50 = 12900 nM T83145 CL59MP 86294771 IC50 = 12900 nM T83145 C4A0EX 90643506 IC50 = 10000 nM T83145 C2BR1Z 90643507 IC50 = 68400 nM T83145 CU6E0X 90644814 IC50 = 16800 nM T83145 CPJ21F 90665954 IC50 = 150 nM T83145 C3KRH8 90665955 IC50 = 62 nM T83145 C1BA4E 90665956 IC50 = 62 nM T83145 CY80KV 90665957 IC50 = 23 nM T83145 CA48LV 90665958 IC50 = 12 nM T83145 CYB86O 90665959 IC50 = 32 nM T83145 CW8MS4 90665960 IC50 = 22 nM T83145 CQ67SO 90665961 IC50 = 25 nM T83145 CN94OJ 90665962 IC50 = 9 nM T83145 C2K9LZ 90665963 IC50 = 38 nM T83145 C81TAL 90665964 IC50 = 110 nM T83145 CP5S0X 90665965 IC50 = 18 nM T83145 C8IVK5 90665966 IC50 = 39 nM T83145 C7DL5F 90665967 IC50 = 17 nM T83145 C78ZBE 90665968 IC50 = 10 nM T83145 C2AG7C 90665969 IC50 = 9 nM T83145 C10CYW 90665970 IC50 = 12 nM T83145 CHBL08 90665971 IC50 = 950 nM T83145 CVZO36 90665972 IC50 = 140 nM T83145 C5EN3W 90665973 IC50 = 320 nM T83145 C62YEW 90665974 IC50 = 120 nM T83145 CQE72G 90665976 IC50 = 53 nM T83145 CYF9H8 90665977 IC50 = 110 nM T83145 CEJL79 90675811 IC50 = 43500 nM T83145 CX8NM0 90675812 IC50 = 12300 nM T83145 C1FH4W 90675813 IC50 = 27900 nM T83145 C5VHX9 90675815 IC50 = 96700 nM T83145 CA2DJ6 90675816 IC50 = 63800 nM T83145 CZE5B2 90675818 IC50 = 44500 nM T83145 CQB9Z3 90675819 IC50 = 26500 nM T83145 CVYO20 90675822 IC50 = 56300 nM T83145 CM8D7J 90675823 IC50 = 48600 nM T83145 C3L8KC 90675826 IC50 = 56300 nM T83145 C3DJA8 90675827 IC50 = 14600 nM T83145 CZDF50 90675829 IC50 = 27100 nM T83145 C2QE0X 90675830 IC50 = 25900 nM T83145 CS89VL 90677190 IC50 = 17500 nM T83145 CY68XI 90681063 IC50 = 11000 nM T83145 CE1T7P 90681064 IC50 > 30000 nM T83145 CBV1X5 90681065 IC50 = 3000 nM T83145 CCS30Q 90681066 IC50 = 8000 nM T83145 C5ZMG1 90681067 IC50 = 12000 nM T83145 CXIT14 90681068 IC50 > 30000 nM T83145 C4YEF9 90681069 IC50 = 13000 nM T83145 CE51CR 90681070 IC50 = 18000 nM T83145 CZK03A 90681071 IC50 > 30000 nM T83145 C1DTR6 90681072 IC50 > 30000 nM T83145 CMB68I 90681073 IC50 = 2800 nM T83145 C0UNZ5 90681074 IC50 = 1200 nM T83145 CHY87P 90681075 IC50 > 30000 nM T83145 CW2E1V 90681076 IC50 > 30000 nM T83145 CU8ZP2 90681746 EC50 = 8270 nM T83145 C4P9LZ 118708694 IC50 = 1940 nM T83145 CC8W2Z 118708695 IC50 = 1800 nM T83145 CMP30W 118708696 IC50 = 2320 nM T83145 CED6Q4 118708697 IC50 = 2040 nM T83145 CK1C7G 118708698 IC50 = 1640 nM T83145 C3T1DS 118708699 IC50 = 740 nM T83145 CB82CY 118708700 IC50 = 960 nM T83145 CE59BN 118708701 IC50 = 820 nM T83145 C7MHC8 118708702 IC50 = 3120 nM T83145 C7T5WJ 118708703 IC50 = 2820 nM T83145 CH8YJ4 118708704 IC50 = 3120 nM T83145 CEY30J 118708705 IC50 > 10000 nM T83145 CD74KN 118712697 IC50 = 4700 nM T83145 C2OM4D 118712698 IC50 = 6900 nM T83145 C5XUW6 118712699 IC50 = 39800 nM T83145 CW5AC6 118716125 IC50 = 500 nM T83145 CK4VQ0 118716126 IC50 > 10000 nM T83145 C48PKT 118716127 IC50 > 10000 nM T83145 CH1OL7 118716128 IC50 = 10000 nM T83145 CQ45JC 118716129 IC50 = 13000 nM T83145 CQ6G7M 118716130 IC50 = 24000 nM T83145 CPY16H 118716131 IC50 = 4200 nM T83145 C0UA6E 118716132 IC50 = 8000 nM T83145 CVRK59 118716133 IC50 = 10000 nM T83145 CVZ56P 118716134 IC50 = 1300 nM T83145 C5P0LJ 118716135 IC50 = 830 nM T83145 CB1AL4 118716136 IC50 = 760 nM T83145 CNZ3P8 118729822 IC50 = 18.2 ug.mL-1 T83145 CSB0M9 135494223 IC50 = 29800 nM T83145 CST9B8 136244569 IC50 = 30000 nM T83145 CSK95Y 136504263 IC50 > 50000 nM T83145 CR2S0C 108068 IC50 = 3400 nM T83145 D0B0IJ 65351 IC50 = 34500 nM T83145 D0EW3L 5281222 IC50 = 38000 nM T83145 D0HD2G 4788 IC50 = 41000 nM T83145 D0IO0I 6474893 IC50 = 1800 nM T83145 D0L2XO 5353431 IC50 = 2000 nM T79473 CUR6Q3 2741928 IC50 = 378 nM T79473 C5ROY0 9887381 EC50 = 220 nM T79473 CJW79C 9915237 Ki = 0.311 nM T79473 C1KI7W 11502667 EC50 = 1500 nM T79473 C2RPC4 11509369 EC50 = 1200 nM T79473 CG42JP 11531195 EC50 = 1900 nM T79473 COQ05A 11539288 EC50 = 800 nM T79473 CHU3C6 11618319 EC50 = 1100 nM T79473 CB1UE5 11654606 EC50 = 800 nM T79473 CRXO16 29993669 IC50 = 403 nM T79473 CY5P9C 29993670 IC50 = 6790 nM T79473 CLVX83 44255904 EC50 = 5 nM T79473 C1UIB6 44440746 EC50 = 250 nM T79473 C8UY9K 44440747 EC50 > 100000 nM T79473 C4SQV6 44440748 EC50 = 500 nM T79473 CTW5P8 44440749 EC50 > 100000 nM T79473 CVQ2S9 44440750 EC50 = 12100 nM T79473 CV2F9O 44440751 EC50 = 170 nM T79473 CS93BX 44440752 EC50 = 150 nM T79473 C0ND3F 44440753 EC50 = 190 nM T79473 CC2V0G 44440754 EC50 = 80 nM T79473 CN5GR8 44440784 EC50 = 2300 nM T79473 CO3TW7 44572264 EC50 = 1600 nM T79473 C4G8NW 53318121 EC50 = 57 nM T79473 C7WMT6 53320758 EC50 = 43 nM T79473 C38TJY 53320759 EC50 = 24 nM T79473 CJ3FE8 53320760 EC50 = 80 nM T79473 C15NUY 53320793 EC50 = 10 nM T79473 CH4JK8 53322111 EC50 = 1 nM T79473 C0JQI4 53323417 EC50 = 27 nM T79473 CQR37K 53324741 EC50 = 75 nM T79473 C2Q3EJ 53324742 EC50 = 61 nM T79473 C1Q5IF 53324743 EC50 = 55 nM T79473 C2S6FJ 53324744 EC50 = 39 nM T79473 CJW08H 57325683 IC50 = 95 nM T79473 CG2NH6 139600336 IC50 = 185 nM T79473 C0HN5J 139600337 IC50 = 97 nM T79473 C4VS6A 155510420 IC50 > 16000 nM T79473 CZP12C 155516839 IC50 = 174 nM T79473 C5K8VI 155520123 IC50 > 16500 nM T79473 CF6I8H 155524816 IC50 = 1680 nM T79473 CLP3I4 155526147 IC50 > 16500 nM T79473 CI0T7H 155527311 IC50 = 81 nM T79473 C8PS0G 155528786 IC50 = 193 nM T79473 CV9C3X 155529559 IC50 > 16500 nM T79473 C9GB8O 155530584 IC50 = 1850 nM T79473 CB8AY3 155530808 IC50 > 16500 nM T79473 CA2Q7T 155532999 IC50 = 2610 nM T79473 CC6FA8 155533073 IC50 = 3650 nM T79473 C8X9FY 155534855 IC50 = 7470 nM T79473 CO6YZ2 155535600 IC50 = 3320 nM T79473 C5JK6F 155542952 IC50 = 207 nM T79473 C6FQW0 155546314 IC50 = 127 nM T79473 CDRE25 155555227 IC50 = 2310 nM T79473 CG28KL 155555948 IC50 = 312 nM T79473 C9K8XW 155558589 IC50 = 1620 nM T79473 CZN94G 155559372 IC50 > 16500 nM T79473 CA0U2G 155561384 IC50 = 275 nM T79473 C2FHL1 155561534 IC50 = 580 nM T79473 CL9P1F 155563159 IC50 = 107 nM T79473 C1DHB3 155563505 IC50 = 5180 nM T79473 CW91NA 155564366 IC50 = 3240 nM T79473 CHC34Z 155565197 IC50 = 332 nM T79473 CLQJ13 155566723 IC50 = 102 nM T79473 C6O0CD 155567488 IC50 = 3130 nM T79473 CKLF48 155568207 IC50 = 486 nM T24548 C5M7RV 130737 Ki = 140 nM T24548 C1DX5A 10262492 Ki = 3100 nM T24548 C8FEI2 44380269 Ki = 5070 nM T68208 CC5Q0Y 73354735 IC50 = 496 nM T68208 CH7GY0 73354736 IC50 = 2003 nM T68208 D05LMD 16134896 IC50 = 266 nM T30985 D02DPA 2756 Ki = 70 nM T30985 D03WEX 9966051 Ki = 180 nM T30985 D04USC 774 EC50 = 463 nM T30985 D0CQ0Z 33630 Ki = 1000 nM T30985 D0G8NN 119570 Ki = 2683 nM T30985 D07YGH 9976892 Ki > 3162.28 nM T30985 D0LI1C 44469321 IC50 > 10000 nM T30985 D0M9RQ 11697697 IC50 > 10000 nM T30985 D0OW9L 11973780 IC50 > 10000 nM T30985 D02KAF 10103168 EC50 = 2500 nM T30985 D05FYA 3035905 Ki > 10000 nM T30985 D0B4TT 17747460 IC50 = 10000 nM T30985 CMD1L2 5818 EC50 = 1258.93 nM T30985 C5H9CN 9287 Ki > 10000 nM T30985 C2VQH8 29298 Ki = 10131 nM T30985 C2VRP9 182527 EC50 = 2570.4 nM T30985 CYP7U8 409544 Ki = 12589.25 nM T30985 CQZ4A9 636934 Ki > 10000 nM T30985 CL3BA9 3201696 IC50 > 20000 nM T30985 C0YXV3 3676358 Ki > 10000 nM T30985 CK4G9W 5250783 Ki = 19952.62 nM T30985 CJ0M1D 9802248 IC50 = 9105 nM T30985 C8XGV3 9804849 IC50 = 860 nM T30985 C5Z2KM 9805944 Ki = 1.7 nM T30985 CIH80R 9818650 Ki = 3781 nM T30985 CEOI07 9822631 IC50 = 1774 nM T30985 CC3RA7 9823337 IC50 > 10000 nM T30985 CT5M1L 9851785 Ki > 10000 nM T30985 CQ4LC2 9872676 Ki = 1220 nM T30985 C34AHG 9880208 Ki = 16982.44 nM T30985 C98ISM 9889247 IC50 = 123 nM T30985 C4NOK6 9889248 IC50 = 691 nM T30985 CYWQ50 9906447 Ki = 1708 nM T30985 CWQ75J 9923147 Ki = 7413.1 nM T30985 CI3V0F 9923186 Ki = 19054.61 nM T30985 C5LW8I 9932752 IC50 = 10000 nM T30985 C3D6KB 9974306 Ki = 1584.89 nM T30985 CXC14J 9979651 IC50 > 10000 nM T30985 CN43CY 9990475 Ki = 10000 nM T30985 CY23MC 10003369 IC50 > 10000 nM T30985 C3YB9L 10003483 Ki = 1800 nM T30985 CJ01QT 10015196 Ki = 5011.87 nM T30985 CE6MC9 10017820 Ki = 1584.89 nM T30985 CP7BX9 10039772 Ki = 12589.25 nM T30985 CMUW84 10064805 Ki = 1729 nM T30985 CP08FW 10069595 Ki = 10232.93 nM T30985 CZ12NX 10085839 Ki = 3981.07 nM T30985 C3IKD4 10138404 IC50 = 10000 nM T30985 C37JZT 10139591 IC50 = 1500 nM T30985 CAC2V4 10139592 IC50 = 870 nM T30985 C9YE7Q 10140544 IC50 = 2100 nM T30985 C0XW3H 10141470 IC50 = 1858 nM T30985 CYON75 10161929 IC50 = 4517 nM T30985 CQ0F2D 10162727 IC50 = 3000 nM T30985 C2S8CB 10202996 IC50 = 1334 nM T30985 CB20RT 10204866 IC50 = 500 nM T30985 CT0DH4 10205121 IC50 = 10000 nM T30985 CGMA86 10226501 IC50 = 3200 nM T30985 CS6MU7 10268636 Ki = 10000 nM T30985 C5Y6MR 10273238 IC50 = 630 nM T30985 CI38FT 10279311 IC50 = 3059 nM T30985 C19KRM 10298838 IC50 = 2900 nM T30985 CN1Y6Z 10341609 Ki = 19498.45 nM T30985 CGOE95 10343536 Ki = 1600 nM T30985 C6M8ZW 10422468 Ki = 10000 nM T30985 C70ZTF 10451094 Ki = 100000 nM T30985 CM8PV0 10455457 Ki = 17782.79 nM T30985 CA76BD 10466840 Ki = 10000 nM T30985 CRM27I 10472082 Ki = 9120.11 nM T30985 CI7D9Z 10473209 Ki > 3162.28 nM T30985 CAZ58C 10478188 IC50 = 5350 nM T30985 CRI50E 10885636 IC50 = 1030 nM T30985 CX65PW 10907460 IC50 = 757 nM T30985 CF15CY 10986211 EC50 > 0.0001 nM T30985 CJC9K4 11005810 IC50 = 368 nM T30985 CG41BK 11071079 IC50 = 1250 nM T30985 CO81WF 11094685 EC50 > 0.0001 nM T30985 C7DE0U 11113605 IC50 = 1340 nM T30985 CWE5L2 11116130 EC50 > 0.0001 nM T30985 CUF10O 11126319 EC50 > 0.0001 nM T30985 CK9N0C 11166846 IC50 = 225 nM T30985 CAX76O 11189839 IC50 = 2150 nM T30985 C4ED6S 11202401 IC50 = 950 nM T30985 C3P9VF 11211919 IC50 = 3050 nM T30985 CL94YG 11212029 IC50 = 3850 nM T30985 CRO3N6 11238716 IC50 = 500 nM T30985 C5ZU6K 11247290 IC50 = 5600 nM T30985 CWSN57 11247939 IC50 = 3100 nM T30985 C1AHS5 11259138 IC50 = 3982 nM T30985 CV6G3A 11282005 IC50 = 3272 nM T30985 CK5P6Q 11293983 IC50 = 260 nM T30985 CAR34I 11328514 IC50 = 850 nM T30985 CRA7Y4 11329753 IC50 = 1397 nM T30985 C3RD1M 11329754 IC50 = 1500 nM T30985 C39RTK 11338659 IC50 > 10000 nM T30985 C6M9XH 11340290 IC50 = 779 nM T30985 CC13FL 11349921 IC50 > 10000 nM T30985 C6TO3F 11351801 IC50 = 6700 nM T30985 CDHE37 11362693 IC50 = 1185 nM T30985 C9AC7J 11363750 IC50 = 5600 nM T30985 CL4WV9 11373970 IC50 > 10000 nM T30985 C6DW4X 11385692 IC50 = 880 nM T30985 C5ZHK8 11393516 Ki = 7762.47 nM T30985 CKQ40V 11396873 IC50 = 500 nM T30985 C85LYP 11430418 IC50 > 1000 nM T30985 C70QJL 11430513 IC50 = 2095 nM T30985 CH8JN4 11443495 IC50 = 2900 nM T30985 CI69YB 11453538 IC50 < 100 nM T30985 CLN5R1 11476077 IC50 = 1915 nM T30985 CI8O3H 11487026 IC50 > 10000 nM T30985 C8GZ1I 11539020 IC50 > 10000 nM T30985 CQ08DH 11539632 IC50 = 0.87 nM T30985 C9UG2V 11544758 Ki > 4000 nM T30985 CE0U8J 11581337 IC50 > 10000 nM T30985 C0G6PN 11632103 IC50 > 10000 nM T30985 CBA3V4 11723317 Ki = 3162.28 nM T30985 C7PVL8 11730467 IC50 = 1980 nM T30985 CW6O3K 11785584 IC50 = 1025 nM T30985 CMDT64 11804748 EC50 > 0.0001 nM T30985 C4JIZ5 11829635 EC50 = 93 nM T30985 C0X7FJ 11846300 Ki = 8709.64 nM T30985 CXLW54 11948707 Ki = 2126 nM T30985 CEI40N 11954293 Ki = 5.7 nM T30985 C8JQL7 11957735 IC50 > 10000 nM T30985 CJ8K3O 12016525 Ki = 41686.94 nM T30985 CNY71B 12192007 Ki = 19054.61 nM T30985 C2X3UC 13170764 EC50 = 1288.25 nM T30985 CT6AL1 16061961 Ki > 1000 nM T30985 CV36OS 16082828 EC50 > 10000 nM T30985 CHTO30 16082831 EC50 > 10000 nM T30985 CJ1DV9 16082833 EC50 > 10000 nM T30985 C08XJA 16718567 IC50 > 30000 nM T30985 C6L3IF 18539962 Ki = 14454.4 nM T30985 CV0EI2 18672441 Ki = 67608.3 nM T30985 C3T5HF 21509921 Ki = 81 nM T30985 CT7XG9 21830793 Ki = 2126 nM T30985 C3BP7D 23151209 IC50 > 10000 nM T30985 CY21RE 24841480 Ki = 540 nM T30985 CZPW63 24936097 Ki > 1000 nM T30985 CQ52SD 24936098 Ki > 1000 nM T30985 C2G1JK 25053351 Ki > 10000 nM T30985 C51OJR 25099115 IC50 > 10000 nM T30985 CMX36H 25107505 Ki > 10000 nM T30985 C7NJ1B 25109291 Ki > 9120.11 nM T30985 CML6G5 25128822 Ki = 31622.78 nM T30985 C8D7HZ 25149335 EC50 = 63.1 nM T30985 CQ7N3X 25149521 EC50 = 78 nM T30985 C92NXM 25149613 EC50 = 120 nM T30985 C4GC8J 25149708 EC50 = 109 nM T30985 C6NAC0 25149712 EC50 = 63.1 nM T30985 CJ1Z9H 25216680 Ki > 10000 nM T30985 C1T3LR 25218143 Ki > 10000 nM T30985 CPI03N 25218397 Ki > 55000 nM T30985 CL1R3Q 25218401 Ki > 10000 nM T30985 CMKQ63 42625221 EC50 = 81.28 nM T30985 CIJ52Y 42625222 EC50 = 954.99 nM T30985 CR7LN9 42625223 EC50 = 346.74 nM T30985 C5O9XR 42625224 EC50 = 30.2 nM T30985 C8G7QX 42625303 EC50 = 371.54 nM T30985 C75WJN 42625304 EC50 = 109.65 nM T30985 C0BW6J 42625384 EC50 = 724.44 nM T30985 CID4J1 42625386 EC50 = 141.25 nM T30985 C5YR2D 42626109 EC50 = 36.31 nM T30985 C4W5PM 42626110 EC50 = 288.4 nM T30985 CI34UC 42626111 EC50 = 83.18 nM T30985 C8P2LE 44250288 IC50 > 10000 nM T30985 CEL7B6 44275464 Ki < 1905.46 nM T30985 CE20CZ 44275807 Ki = 10000 nM T30985 CA0DN5 44304003 Ki = 72443.6 nM T30985 C3Z5DG 44304012 Ki = 40738.03 nM T30985 CZ5X0G 44304013 Ki = 19054.61 nM T30985 CK63QN 44304014 Ki = 45708.82 nM T30985 C1P7BD 44304021 Ki = 21877.62 nM T30985 CNKS56 44304030 Ki = 20417.38 nM T30985 CJF2S5 44304031 Ki = 6760.83 nM T30985 CK7Q8R 44304032 Ki = 27542.29 nM T30985 CGA15P 44304035 Ki = 12589.25 nM T30985 CY2JQ9 44304036 Ki = 22387.21 nM T30985 CGP5R0 44304037 Ki = 22387.21 nM T30985 C6D4QK 44304049 Ki = 24547.09 nM T30985 C95EPL 44304056 Ki = 50118.72 nM T30985 C8FUS4 44304064 Ki = 33113.11 nM T30985 CTZB24 44304066 Ki = 17782.79 nM T30985 C1I2VN 44304067 Ki = 79432.82 nM T30985 C7BOY8 44304068 Ki = 20417.38 nM T30985 CS7V9L 44304079 Ki = 69183.1 nM T30985 CCH2E6 44304088 Ki = 7943.28 nM T30985 C9IM6V 44304090 Ki = 79432.82 nM T30985 CY0SG5 44304091 Ki = 2691.53 nM T30985 CP3DB1 44304211 Ki = 10964.78 nM T30985 CL9F2Z 44304223 Ki = 9549.93 nM T30985 CP0Z1H 44304243 Ki = 7585.78 nM T30985 CU6LJ1 44304244 Ki = 18620.87 nM T30985 CQ86HY 44304245 Ki = 11748.98 nM T30985 CY5NQ8 44304246 Ki = 12882.5 nM T30985 CKE47A 44304247 Ki = 19952.62 nM T30985 CG5TJ8 44304256 Ki = 27542.29 nM T30985 C1GQH4 44304259 Ki = 19498.45 nM T30985 C4RL7Y 44304269 Ki = 22387.21 nM T30985 CLH2M5 44304270 Ki = 8128.31 nM T30985 C2RPN4 44304277 Ki = 48977.88 nM T30985 CVXS65 44304282 Ki = 3715.35 nM T30985 C0A8SI 44304283 Ki = 1548.82 nM T30985 C6G3YS 44304284 Ki = 8317.64 nM T30985 CQU2W4 44304287 Ki = 14791.08 nM T30985 CYX69C 44304288 Ki = 31622.78 nM T30985 CUN8B6 44304291 Ki = 29512.09 nM T30985 CK5OM8 44304293 Ki = 15135.61 nM T30985 C9U0HX 44304294 Ki = 20892.96 nM T30985 CC76QK 44304295 Ki = 10000 nM T30985 CSR0G4 44304303 Ki = 12302.69 nM T30985 CBH73L 44304304 Ki = 25118.86 nM T30985 C97BJW 44304307 Ki = 22908.68 nM T30985 CHR62F 44304308 Ki = 17378.01 nM T30985 CUWM24 44304309 Ki = 42657.95 nM T30985 C1J2NZ 44304310 Ki = 14791.08 nM T30985 CFSR60 44304311 Ki = 97723.72 nM T30985 C13YKA 44304312 Ki = 39810.72 nM T30985 CJ0DI3 44304313 Ki = 46773.51 nM T30985 CZ1RI6 44304316 Ki = 50118.72 nM T30985 C5W1TM 44304318 Ki = 10232.93 nM T30985 CJY49E 44304319 Ki = 10715.19 nM T30985 C3YC4E 44304320 Ki = 10715.19 nM T30985 C7RJ8O 44304325 Ki = 23442.29 nM T30985 CVT19R 44304327 Ki = 10000 nM T30985 CBJK06 44304329 Ki = 53703.18 nM T30985 C3B0GW 44304331 Ki = 10000 nM T30985 C3-FEB-02 44304332 Ki = 89125.09 nM T30985 C6J5OZ 44304348 Ki = 60255.96 nM T30985 CN2W8Q 44304349 Ki = 14791.08 nM T30985 CC9PT2 44304357 Ki = 57543.99 nM T30985 CSX2L0 44304376 Ki = 18620.87 nM T30985 CEWD86 44304377 Ki = 46773.51 nM T30985 CZ86DV 44304378 Ki = 60255.96 nM T30985 C0TYR3 44304382 Ki = 11220.18 nM T30985 CH23XB 44304383 Ki = 3715.35 nM T30985 CP7I3Z 44304385 Ki = 17782.79 nM T30985 C7ZF0Q 44304387 Ki = 39810.72 nM T30985 CV3O9C 44304393 Ki = 12589.25 nM T30985 CZ0Q7N 44304399 Ki = 1862.09 nM T30985 CEQO51 44304402 Ki = 7079.46 nM T30985 CT7L5H 44304412 Ki = 13489.63 nM T30985 C1KIA2 44304415 Ki = 22908.68 nM T30985 COP9L3 44304431 Ki = 12022.64 nM T30985 CS20NC 44304437 Ki = 24547.09 nM T30985 CV7U0X 44304438 Ki = 22908.68 nM T30985 C9OES6 44304439 Ki = 8912.51 nM T30985 C4KX8A 44304445 Ki = 3467.37 nM T30985 CKY4V8 44304449 Ki = 4466.84 nM T30985 CF2X5I 44304450 Ki = 38018.94 nM T30985 C95OLE 44304451 Ki = 31622.78 nM T30985 C5I2QL 44304457 Ki = 12022.64 nM T30985 CB6G5H 44304459 Ki = 2137.96 nM T30985 C6JT1P 44304462 Ki = 34673.69 nM T30985 CUR3O7 44304475 Ki = 56234.13 nM T30985 C19UMQ 44304494 Ki = 10715.19 nM T30985 CQ6A4T 44304516 Ki = 26915.35 nM T30985 CMGY49 44304558 Ki = 31622.78 nM T30985 CX97UN 44304560 Ki = 14125.38 nM T30985 CO6ZF2 44304719 Ki = 89125.09 nM T30985 CR2YO1 44304741 Ki = 34673.69 nM T30985 C57WXT 44304743 Ki = 16595.87 nM T30985 CN51UA 44304751 Ki = 12302.69 nM T30985 CP05OY 44304752 Ki = 83176.38 nM T30985 CNEK74 44304753 Ki = 37153.52 nM T30985 CE6P5V 44304760 Ki = 14125.38 nM T30985 C6WM1H 44304978 Ki = 83176.38 nM T30985 C5OYK1 44304990 Ki = 12302.69 nM T30985 CDHT79 44304991 Ki = 20892.96 nM T30985 CT63YZ 44307779 Ki = 3211 nM T30985 CG6Z4H 44333987 Ki = 24000 nM T30985 CA7OE5 44333988 Ki = 3500 nM T30985 CGR23Y 44334025 Ki = 1000 nM T30985 C46JFI 44334035 Ki = 4000 nM T30985 C9MFY5 44334036 Ki = 6100 nM T30985 CZ9LJ8 44334037 Ki = 6200 nM T30985 C37JOG 44334038 Ki = 900 nM T30985 C2L8JG 44334042 Ki = 710 nM T30985 CJ96XL 44334212 Ki = 330 nM T30985 CGPL96 44334214 Ki = 2300 nM T30985 CJB65X 44334234 Ki = 7100 nM T30985 C13TRB 44334235 Ki = 2200 nM T30985 C9PY0X 44334252 Ki = 100000 nM T30985 CY8XM2 44334265 Ki = 5000 nM T30985 CP4W5X 44334281 Ki = 40000 nM T30985 C9BS4V 44334368 Ki = 290 nM T30985 CM57UH 44334369 Ki = 730 nM T30985 C9M1NZ 44334395 Ki = 500 nM T30985 C1EQY2 44334396 Ki = 1550 nM T30985 CC1RW3 44334406 Ki = 290 nM T30985 C18SHG 44334407 Ki = 700 nM T30985 CDQ72F 44334430 Ki = 1200 nM T30985 CS7YO0 44334503 Ki = 22000 nM T30985 CM15VJ 44334521 Ki = 31000 nM T30985 CFHU75 44334556 Ki = 46000 nM T30985 C9XC5R 44334781 Ki = 1000 nM T30985 CXD0C7 44334782 Ki = 380 nM T30985 C1L3GT 44335172 Ki = 97723.72 nM T30985 C6KCD9 44335185 Ki = 1659.59 nM T30985 C24HSP 44335222 Ki = 57543.99 nM T30985 C4BLC5 44335225 Ki = 12302.69 nM T30985 C8HYU5 44335237 Ki = 3981.07 nM T30985 C1TL7P 44335238 Ki = 23988.33 nM T30985 C51LMP 44335336 Ki = 33884.42 nM T30985 C7R2BK 44335350 Ki = 100000 nM T30985 CDFA49 44335351 Ki = 5623.41 nM T30985 CCY4I9 44335368 Ki = 23988.33 nM T30985 CCI26P 44335384 Ki = 18620.87 nM T30985 CNF4S6 44335387 Ki = 28840.32 nM T30985 CO75LT 44335389 Ki = 7585.78 nM T30985 C2ZN6D 44335405 Ki = 22908.68 nM T30985 C18ONA 44335407 Ki = 3630.78 nM T30985 C7LH1C 44335412 Ki = 8317.64 nM T30985 C89TNO 44335428 Ki = 69183.1 nM T30985 CPQW41 44335430 Ki = 33113.11 nM T30985 C04MTD 44335456 Ki = 10000 nM T30985 CO0GR9 44335463 Ki = 12882.5 nM T30985 CMD1U0 44335483 Ki = 12882.5 nM T30985 C12MNS 44335558 Ki = 9120.11 nM T30985 CJX50C 44335559 Ki = 11748.98 nM T30985 CN9JI6 44335571 Ki = 38018.94 nM T30985 CF8GV3 44414337 EC50 = 160 nM T30985 CZL97F 44455426 Ki = 3178 nM T30985 C7UDS1 44467360 Ki = 4900 nM T30985 CQ0WM7 44469273 IC50 > 5000 nM T30985 C4DL5C 44469677 IC50 > 10000 nM T30985 CK10AW 44478385 Ki = 4073.8 nM T30985 CJ27OY 44480707 EC50 = 7244.36 nM T30985 C37FDB 44481214 EC50 = 1995.26 nM T30985 CB9E6J 44481217 EC50 = 12022.64 nM T30985 CDX0I8 44481485 EC50 > 10000 nM T30985 CL91FN 44481487 EC50 = 3890.45 nM T30985 C3SJ9D 44481489 EC50 = 14125.38 nM T30985 CO26SI 44481758 EC50 = 8912.51 nM T30985 C98MAW 44482299 EC50 = 436.52 nM T30985 CJ2ST3 44482300 EC50 = 380.19 nM T30985 CT82CQ 44482302 EC50 = 12022.64 nM T30985 CVA67X 44568347 Ki = 1400 nM T30985 CRCH48 44582675 Ki = 2428 nM T30985 CEJ4R8 44582676 Ki = 1757 nM T30985 C5QB4K 44582678 Ki = 1156 nM T30985 C01RCI 44582705 Ki = 827 nM T30985 CYXD79 45257131 Ki > 1000 nM T30985 C07WHQ 45257132 Ki > 1000 nM T30985 CY25IH 45257133 Ki > 1000 nM T30985 C3QU2C 45487384 IC50 > 5000 nM T30985 CU15OL 46235428 EC50 > 10000 nM T30985 CN75IJ 46830167 EC50 = 79.43 nM T30985 CK8A1O 46880462 Ki > 10000 nM T30985 C9KDP4 46880463 Ki > 10000 nM T30985 CODR73 46880498 Ki > 10000 nM T30985 CHJ5Y6 46880566 Ki > 10000 nM T30985 CE9PG2 46880567 Ki > 10000 nM T30985 C01PGO 46880568 Ki > 10000 nM T30985 CS7L4X 46880569 Ki > 10000 nM T30985 C0PXY7 46880628 Ki > 10000 nM T30985 CD37LU 46880629 Ki > 10000 nM T30985 CUY89F 46880630 Ki > 10000 nM T30985 C4P6XS 46880631 Ki > 10000 nM T30985 CJ53KF 46880672 Ki > 10000 nM T30985 CYJC08 46880673 Ki > 10000 nM T30985 C1RI9O 46880674 Ki > 10000 nM T30985 CL6Z7Q 46884734 Ki = 4.5 nM T30985 CB29TI 46887041 EC50 = 120.23 nM T30985 C9P3CV 46887042 EC50 = 18.62 nM T30985 C12SYH 46887043 EC50 = 6.457 nM T30985 CQJ8W2 46887076 EC50 = 50.12 nM T30985 CAG89L 46887077 EC50 = 53.7 nM T30985 COK81L 46887078 EC50 = 28.18 nM T30985 CB09SD 46887079 EC50 = 9.333 nM T30985 CK0S2U 46887080 EC50 = 20.42 nM T30985 CLPJ52 46887115 EC50 = 28.84 nM T30985 COR71G 46890166 EC50 = 131 nM T30985 C8FR9E 46890592 EC50 > 10000 nM T30985 CDV30W 46912441 Ki > 1000 nM T30985 CAQ0E9 46912442 Ki > 1000 nM T30985 C6F2MP 46929551 Ki > 10000 nM T30985 CT3UX6 46929553 Ki > 10000 nM T30985 CZJ2G8 46929554 Ki > 10000 nM T30985 C40EGB 46929647 Ki > 10000 nM T30985 CB95RA 46929648 Ki > 10000 nM T30985 C2RY0J 50878551 Ki = 4247 nM T30985 C1W6TV 50898777 Ki = 3162.28 nM T30985 CXMZ73 50898778 Ki > 10000 nM T30985 CE4KP1 51050257 Ki > 10000 nM T30985 CODA90 53320569 Ki = 2148 nM T30985 C32YWL 53324045 Ki = 278 nM T30985 CR4W9L 53324553 Ki = 4423 nM T30985 CRQF15 53325242 Ki = 546 nM T30985 CB37XF 53325861 Ki = 4450 nM T30985 CMOZ61 53475319 Ki = 224 nM T30985 CB72FX 54754351 Ki = 3560 nM T30985 CPS5V6 54764158 Ki > 10000 nM T30985 CY92VU 56835087 Ki > 10000 nM T30985 C0JMA7 56835088 Ki > 10000 nM T30985 C1MIQ2 56953887 EC50 = 57.54 nM T30985 CEV7F6 56953889 EC50 = 47.86 nM T30985 CGU3D8 56953998 EC50 = 44.67 nM T30985 C8ZT0L 56954000 EC50 = 7.762 nM T30985 C46SBY 56954002 EC50 = 16.6 nM T30985 CUKA84 56954125 EC50 = 25.7 nM T30985 CEG0H8 56954129 EC50 = 30.9 nM T30985 CQ4AG3 56954227 EC50 = 21.38 nM T30985 C36MDB 56954229 EC50 = 93.33 nM T30985 C7B8RI 56954318 EC50 = 213.8 nM T30985 C7G3TI 56954320 EC50 = 56.23 nM T30985 CKG35O 56954322 EC50 = 6.166 nM T30985 CI7XO6 56954425 EC50 = 24.55 nM T30985 CGVI36 56954513 EC50 = 13.8 nM T30985 CIQH95 56954515 EC50 = 7.586 nM T30985 CWEB27 56954517 EC50 = 151.36 nM T30985 C1TC7Q 56963799 Ki = 923 nM T30985 CI5M2U 57395620 Ki = 8820 nM T30985 C4RHF3 57404027 Ki > 10000 nM T30985 CUOV05 57411066 Ki > 10000 nM T30985 CYKF93 59651916 Ki > 10000 nM T30985 CD3U6K 68731121 Ki > 10000 nM T30985 C6IP8Q 69082816 Ki > 10000 nM T30985 CH3SB0 69355600 Ki = 15135.61 nM T30985 CKD60A 70789640 Ki = 443 nM T30985 C6QYO1 71449142 Ki = 6165.95 nM T30985 C6DU5P 71450548 Ki = 9794 nM T30985 CE6YD5 71450707 Ki = 5500 nM T30985 C4TWS5 71452172 Ki = 5157 nM T30985 C4NDR3 71452382 Ki = 400 nM T30985 C6ZWV2 71452383 Ki = 1780 nM T30985 CP45AB 71452695 Ki = 1600 nM T30985 C4X9KY 71454294 Ki = 6100 nM T30985 CA65OQ 71454295 Ki = 530 nM T30985 C6G2HC 71455894 Ki = 3581 nM T30985 CD4HQ6 71456045 Ki > 10000 nM T30985 CD78KL 71456046 Ki = 3200 nM T30985 CSX5J0 71457844 Ki = 4200 nM T30985 C1VOU3 71458814 EC50 = 20.42 nM T30985 CK5T4P 71459604 Ki = 948 nM T30985 CD10CQ 71459761 Ki = 460 nM T30985 CKX5O8 71463061 Ki = 743 nM T30985 C1Y9IC 71463063 Ki = 7267 nM T30985 CRM9Q1 71525678 Ki = 14125.38 nM T30985 C2GK7O 71525679 Ki = 3162.28 nM T30985 C8A0NC 71525681 Ki = 2818.38 nM T30985 CWH6T3 72548703 IC50 = 142 nM T30985 CC6Q5R 72771081 Ki < 100 nM T30985 CC65OA 73213195 Ki > 10000 nM T30985 CW83DK 73213196 Ki = 933.25 nM T30985 CCV91B 73346042 Ki = 1767 nM T30985 CK0HR9 73346334 Ki = 3896 nM T30985 CR97NO 73347825 Ki = 1480 nM T30985 CFW96K 73347828 Ki > 10000 nM T30985 CW8A0Y 73349359 Ki = 1733 nM T30985 C6BS5L 73349361 Ki = 3038 nM T30985 C87LGB 73352415 Ki > 10000 nM T30985 C1NJ0R 73353884 Ki = 1157 nM T30985 C4F7VK 73355415 Ki = 6268 nM T30985 CAI63V 73355417 Ki = 3471 nM T30985 C81CIL 73355418 Ki = 1868 nM T30985 CN5V0R 73355421 Ki = 8517 nM T30985 C2E7QW 75201901 Ki = 8000 nM T30985 C8IDL3 75306277 Ki = 79.43 nM T30985 C98BJM 90643887 IC50 > 10000 nM T30985 CA5Q3N 90667232 EC50 = 239.88 nM T30985 CTF87B 90667234 EC50 = 741.31 nM T30985 CDMQ18 90667235 EC50 = 407.38 nM T30985 CCX29F 90667237 EC50 = 16218.1 nM T30985 CE8MP7 90667262 EC50 = 831.76 nM T30985 CFA3D4 112936251 Ki = 10232.93 nM T30985 C4G3YC 118734875 Ki > 10000 nM T30985 C9AIE1 118734876 Ki > 10000 nM T30985 C7ODW3 122195524 Ki > 900 nM T30985 CM57GR 126720252 Ki = 365 nM T30985 C8MC1I 127028408 Ki = 3388 nM T30985 CR61YN 127034912 Ki < 100 nM T30985 C0Z9RT 127035835 Ki = 6918.31 nM T30985 C4YM3O 127040635 IC50 < 10000 nM T30985 C2XT3K 127048890 EC50 > 10000 nM T30985 CG35RK 127049855 Ki = 9820 nM T30985 C5BZ6T 127049856 Ki = 7360 nM T30985 CF0Y6S 127050431 Ki > 10000 nM T30985 C5P1EB 127050776 Ki > 10000 nM T30985 CH8G4Z 127051047 Ki > 10000 nM T30985 CH8Y7R 127051301 Ki > 10000 nM T30985 CB25IM 127051958 EC50 > 10000 nM T30985 C9OSN3 127052293 Ki = 10300 nM T30985 C3WA2L 127052294 Ki = 7250 nM T30985 C50GOC 130442480 Ki = 8200 nM T30985 CM04RF 130442572 Ki = 6700 nM T30985 CS58HX 132060734 Ki > 10000 nM T30985 CY8B9L 132060743 Ki = 285 nM T30985 C4VNA6 132060746 Ki = 1072 nM T30985 C4OC0I 132060752 Ki = 1099 nM T30985 C7FM0U 132060763 Ki = 985 nM T30985 CGHO19 132060770 Ki = 507 nM T30985 CT81OY 132060776 Ki = 1760 nM T30985 CAVB41 132584404 Ki > 10000 nM T30985 C2OQB5 132609385 IC50 = 1000 nM T30985 CBU81N 134149168 Ki > 10000 nM T30985 C1GY2T 135156251 EC50 > 10000 nM T30985 CBS93O 136030655 Ki > 1000 nM T30985 C8I7CO 136141537 Ki > 1000 nM T30985 CRH19Y 136192874 Ki > 1000 nM T30985 C56FVS 136192886 Ki > 1000 nM T30985 C7FW4R 136239492 Ki > 10000 nM T30985 CPCY48 137645406 Ki = 596 nM T30985 CPI68E 137646281 Ki = 871 nM T30985 CT5CX0 145973771 Ki = 829 nM T30985 C8I7QL 145980875 Ki = 401 nM T30985 CUGO10 145988693 Ki = 252 nM T30985 CCP2U1 145992489 Ki = 526 nM T30985 CC2G1V 146025727 Ki = 2500 nM T30985 C6P3SR 153287553 Ki = 1995.26 nM T30985 CV9G7Z 153287572 Ki > 10000 nM T30985 CO85KL 153287574 Ki > 10000 nM T30985 CGAP59 155512724 Ki > 1000 nM T30985 C20UBG 155513611 Ki > 1000 nM T30985 CU67HI 155513890 Ki = 3640 nM T30985 CTZL14 155516421 Ki > 10000 nM T30985 CGO36Z 155517879 Ki > 1000 nM T30985 CUSA24 155519891 Ki > 10000 nM T30985 C7Y6LX 155523256 EC50 = 245.47 nM T30985 CI2Z8F 155524114 Ki > 10000 nM T30985 CQS1N5 155525278 Ki > 10000 nM T30985 C2K4YP 155525816 EC50 = 75.86 nM T30985 CD4F1G 155531771 Ki = 562.34 nM T30985 C1E5FH 155532722 EC50 = 880 nM T30985 CNK51Q 155535097 Ki > 10000 nM T30985 CB79ZW 155536080 Ki > 10000 nM T30985 C6QN1S 155538988 Ki > 10000 nM T30985 CI37OT 155539096 Ki > 10000 nM T30985 C9S2IA 155539605 Ki = 823 nM T30985 CHQ7A8 155541279 Ki > 10000 nM T30985 C96YSN 155542256 EC50 = 5180 nM T30985 CMT60C 155543832 Ki = 2600 nM T30985 CI5HT7 155544816 EC50 = 2120 nM T30985 C5EV7C 155544839 EC50 = 5290 nM T30985 CO2J0Z 155546798 Ki > 10000 nM T30985 C1T0BF 155549318 Ki > 10000 nM T30985 C0OK3E 155551348 Ki = 6380 nM T30985 C7WO9P 155552060 Ki > 1000 nM T30985 CZQW48 155552101 Ki > 1000 nM T30985 CLK7U1 155552340 Ki > 1000 nM T30985 CF0W4K 155552683 Ki = 520 nM T30985 CMD3T6 155553964 EC50 = 77.62 nM T30985 C2Q6KU 155558968 Ki = 546 nM T30985 CGH2Y1 155559319 EC50 = 95.5 nM T30985 C5BAG2 155559502 Ki > 10000 nM T30985 CQ75DA 155565842 EC50 = 316.23 nM T30985 CHD6C8 155567107 Ki > 1000 nM T30985 CL54XY 155567151 EC50 = 360 nM T30985 C3N9VU 10251906 Ki > 500 nM T30985 CP9TR0 10324985 Ki = 302 nM T30985 D01JXM 46222048 Ki > 1000 nM T30985 D02SQF 37463 EC50 = 2884.03 nM T30985 D05BYD 9906860 Ki = 70794.58 nM T30985 D05RGW 11313837 Ki < 10000 nM T30985 D05ZUX 44207909 Ki >= 1000 nM T30985 D06RNM 3032915 Ki = 3981.07 nM T30985 D09RPR 16737207 Ki > 10000 nM T30985 D0B1KT 15953802 Ki = 100000000 nM T30985 D0B4SF 41376 Ki = 501.19 nM T30985 D0C7LY 11496610 Ki = 850 nM T30985 D0D8GV 9830741 Ki > 1000 nM T30985 D0E5XM 13499360 Ki = 794328.23 nM T30985 D0E7AZ 50287 Ki = 18 nM T30985 D0E9SR 4908365 Ki > 8511.38 nM T30985 D0FF6S 16038374 IC50 > 10000 nM T30985 D0H3DY 10374457 EC50 = 696 nM T30985 D0H4TP 9798547 Ki > 3162.28 nM T30985 D0I3XA 6422124 Ki > 10000 nM T30985 D0I5CT 126688 EC50 = 190.55 nM T30985 D0J6XO 9884746 Ki = 10000 nM T30985 D0KK4C 10154137 EC50 > 0.0001 nM T30985 D0L5MW 181743 Ki = 672 nM T30985 D0M9IC 441082 Ki > 10000 nM T30985 D0O3NG 3077 Ki = 25118.86 nM T30985 D0OM9G 3035842 Ki > 1000 nM T30985 D0SQ0T 10942498 EC50 > 0.0001 nM T30985 D0T2RY 9948320 Ki >= 1000 nM T30985 D0YZ3E 44435200 Ki = 7500 nM T25200 C9AE2B 449135 EC50 = 0.15 nM T25200 CPU83D 503593 EC50 = 0.5 nM T25200 CJ35SZ 703281 EC50 = 22000 nM T25200 CB7ZY9 714750 EC50 = 26000 nM T25200 C5EY7V 827010 EC50 = 22000 nM T25200 CMLS05 1120446 EC50 = 48000 nM T25200 C34VXI 2887294 EC50 = 99000 nM T25200 CO52KZ 2887364 EC50 = 79000 nM T25200 CQTO30 9988610 EC50 = 0.13 nM T25200 CTV8S6 10079983 EC50 = 0.24 nM T25200 CV4S8D 11528282 EC50 = 1000 nM T25200 CL78TG 11528283 EC50 > 1000 nM T25200 C6NZ4F 11542734 EC50 > 1000 nM T25200 CTF46X 11542735 EC50 > 1000 nM T25200 CKZ9I8 11557243 EC50 > 1000 nM T25200 C20LGM 11579082 EC50 = 300 nM T25200 C36JDS 11672622 EC50 = 200 nM T25200 CO0R4C 11679765 EC50 > 1000 nM T25200 CI05CL 11686847 EC50 = 9.7 nM T25200 CXT47O 11708011 EC50 > 1000 nM T25200 CR0Q1L 24810890 EC50 = 90000 nM T25200 C59STH 44278495 IC50 = 2300 nM T25200 C5VF7A 44340439 EC50 = 16 nM T25200 CLW48A 44340440 EC50 = 0.68 nM T25200 CNFJ38 44340441 EC50 = 4 nM T25200 C1XQF7 44340640 EC50 = 0.7 nM T25200 CE8PT9 46230268 EC50 = 2.3 nM T25200 CW8IT2 46230269 EC50 > 50 nM T25200 C9YLJ0 46230270 EC50 > 50 nM T25200 C6Q0PC 46230271 EC50 = 2.5 nM T25200 CP17YX 46874270 IC50 > 50000 nM T25200 CY58UQ 46875163 IC50 = 1000 nM T25200 CFY19G 46875164 IC50 > 50000 nM T25200 C7L2FK 56950527 EC50 = 15 nM T25200 COC45I 56950528 EC50 = 6.5 nM T25200 C2TX6L 56950658 EC50 = 4.2 nM T25200 CN5EW8 70682115 EC50 = 300 nM T25200 CM6C5G 70686402 EC50 = 1000 nM T25200 CAC6R0 70690536 EC50 > 1000 nM T25200 C2TXY8 70692669 EC50 = 1000 nM T25200 C2D4WP 70692681 EC50 > 1000 nM T25200 C4UGR6 70694724 EC50 > 1000 nM T25200 CB8O9M 70696758 EC50 = 53 nM T25200 COH15N 70696759 EC50 = 300 nM T25200 C8BTY5 70696771 EC50 > 1000 nM T25200 CSA5C8 73350701 EC50 = 19.1 nM T25200 CZ3C8S 73350702 EC50 = 6.1 nM T25200 CGBK08 73356728 EC50 = 241 nM T25200 CQU7G9 127048355 EC50 = 20.3 nM T25200 CVAR52 127048361 EC50 = 84 nM T25200 C7T5JU 127048714 EC50 = 0.45 nM T25200 CGR81W 127049706 EC50 = 134 nM T25200 CIDV74 127050308 EC50 = 2.7 nM T25200 CR8L6W 127052457 EC50 = 2.4 nM T25200 C10TYN 135438932 EC50 = 50000 nM T25200 CHU83D 135620685 EC50 = 49000 nM T68320 C82BHU 447280 IC50 = 2900 nM T68320 CB3I6Y 10521264 IC50 > 1000000 nM T68320 CN9M6R 10592387 IC50 = 88000 nM T68320 C8PC9N 10624384 IC50 = 470000 nM T68320 CTSJ57 10665335 IC50 = 2600 nM T68320 CAH46W 10672283 IC50 = 11000 nM T68320 C0YD1X 10687736 IC50 = 30000 nM T68320 CN96PD 11724034 IC50 = 130 nM T68320 C2WUP4 11794649 IC50 = 79000 nM T68320 CS40ML 44123747 IC50 > 50000 nM T68320 C3IS2X 44316877 IC50 = 21000 nM T68320 C6ITG5 44316896 IC50 = 29000 nM T68320 CS02PC 44317216 IC50 = 3400 nM T68320 D0CG7Q 10336627 IC50 = 230 nM T99029 CHGI09 6597 IC50 = 5560000 nM T99029 CMC1D0 12892 Ki = 2851 nM T99029 C6NQ9Y 1116656 IC50 = 5700 nM T99029 CG7X9S 7178546 EC50 = 24500 nM T99029 CKQY13 28361735 IC50 = 8300 nM T99029 C28NIL 29255080 IC50 = 3900 nM T99029 C80ODY 67932020 Ki = 550 nM T99029 CELO13 72376512 IC50 = 21300 nM T99029 C47XUW 86280454 IC50 = 26 nM T99029 CI7HO1 97281116 IC50 = 7800 nM T99029 C3FC0O 126200721 IC50 = 4900 nM T99029 CKQ63N 134561155 IC50 = 1710 nM T99029 C8W3YG 136087021 IC50 = 5336 nM T99029 C0BUJ9 136249185 IC50 = 4800 nM T99029 CI5TH3 137653481 Ki = 2987 nM T99029 C3SV7G 137659540 Ki = 7762 nM T99029 CL6T4P 149986651 IC50 = 59 nM T99029 C24DWX 150179460 IC50 = 461 nM T99029 CJ17UR 150426809 IC50 = 90 nM T99029 C1Z5DA 151004457 IC50 = 5 nM T99029 C02NBO 151026196 IC50 = 67 nM T99029 C0Q9PK 151406722 IC50 = 181 nM T99029 C2RVC3 151777753 IC50 = 255 nM T99029 CKR2T1 151835909 IC50 = 186 nM T99029 CTI5R1 151961601 IC50 = 136 nM T99029 CC3ME1 152131905 IC50 = 80 nM T99029 CAR6N3 152143591 IC50 = 90 nM T99029 C79SKI 152618834 IC50 = 858 nM T99029 C49BFR 155510663 IC50 = 142 nM T99029 CCG7K6 155528322 IC50 = 64 nM T99029 C8EH6M 155538895 IC50 = 98 nM T99029 D0ZA6G 6323491 IC50 = 230000 nM T56697 C93UKS 11617172 EC50 = 7800 nM T56697 CT3XE1 25199517 EC50 = 630 nM T56697 CVNK24 25210880 EC50 = 1000 nM T56697 C9A3ED 25216880 EC50 = 1000 nM T56697 C4AGX2 44550927 EC50 = 9800 nM T56697 C52TUH 44551057 EC50 = 1900 nM T67162 D00KHM 16362 Ki = 11.7 nM T67162 D00TLN 2913 Ki = 112 nM T67162 D01AZG 5073 Ki = 0.44 nM T67162 D01FFA 72301 IC50 = 450 nM T67162 D01ZII 2726 IC50 = 1 nM T67162 D02HED 4748 IC50 = 0.3 nM T67162 D03DJL 6918554 EC50 > 10000 nM T67162 D03ELL 2159 IC50 = 3.04 nM T67162 D03KQF 4011 Ki = 665 nM T67162 D03QGM 5355 Ki = 7.6 nM T67162 D04JCN 47811 Ki = 4 nM T67162 D04JEE 4946 EC50 > 5011.87 nM T67162 D04KJO 3410 IC50 > 10000 nM T67162 D04PHC 5816 Ki = 910 nM T67162 D05DVP 5717 IC50 > 10000 nM T67162 D05MBZ 129211 Ki = 13 nM T67162 D05XGO 11154555 EC50 = 0.4 nM T67162 D05ZIK 4205 Ki > 5454 nM T67162 D06OSM 91273 Ki = 460 nM T67162 D06XZR 27400 Ki = 2.4 nM T67162 D06YFA 31101 Ki = 10 nM T67162 D06ZUK 3696 IC50 = 410 nM T67162 D07MEH 3033769 Ki = 1.21 nM T67162 D07MOX 439260 IC50 = 0.00008 nM T67162 D08VRO 3822 Ki = 240 nM T67162 D0B0CP 667467 Ki = 2.96 nM T67162 D0B3UJ 115237 IC50 = 8.28 nM T67162 D0CQ0Z 33630 Ki = 159 nM T67162 D0D1AL 3559 Ki = 0.12 nM T67162 D0G8NN 119570 Ki = 4.7 nM T67162 D0H3HM 60795 Ki = 0.2 nM T67162 D0H6QU 6005 Ki = 0.62 nM T67162 D0H7KF 5002 Ki = 63.1 nM T67162 D0I0DL 3689 IC50 > 1000 nM T67162 D0I8FI 3779 Ki = 12000 nM T67162 D0J5RN 9690109 IC50 = 2.1 nM T67162 D0KS6W 7077 Ki = 2740 nM T67162 D0L5YV 5152 Ki = 32000 nM T67162 D0M8VE 71360 IC50 = 110 nM T67162 D0O6SX 3658 Ki = 378 nM T67162 D0P0OU 11978813 Ki = 0.3 nM T67162 D0P5SA 3372 Ki = 1.44 nM T67162 D0R1JV 60854 Ki = 0.8 nM T67162 D0R6BI 3341 Ki = 810 nM T67162 D0R6RO 4184 Ki = 2197 nM T67162 D0R9EQ 5095 Ki = 3.7 nM T67162 D0T2XU 4927 IC50 = 100 nM T67162 D0T6QX 5736 Ki = 11 nM T67162 D0T7OW 681 IC50 = 0.000008 nM T67162 D0U1OE 5452 Ki = 27 nM T67162 D0U2OO 2477 Ki = 13 nM T67162 D0U5OE 3964 Ki = 21 nM T67162 D0V4QS 135398745 Ki = 2.1 nM T67162 D0X6BV 6918314 Ki = 666 nM T67162 D0X7KB 28864 Ki = 0.5 nM T67162 D0X7QQ 16363 Ki = 0.027 nM T67162 D0Y5AM 444031 EC50 > 10000 nM T67162 D0Y5UG 2160 Ki = 196 nM T67162 D0Y7XC 5374 Ki = 616.6 nM T67162 D0Z1RV 135398737 Ki = 7.11 nM T67162 D0Z1WA 4916 Ki = 86000 nM T67162 D0Z6UC 5358 Ki > 218 nM T67162 D00POS 9931976 Ki > 50 nM T67162 D01GEB 219050 EC50 = 0.37 nM T67162 D03RIO 24743758 Ki = 251.19 nM T67162 D07YVK 9818479 EC50 = 4.6 nM T67162 D08GJH 125564 Ki = 0.14 nM T67162 D09IRN 21071390 Ki = 1215 nM T67162 D0C8PE 16058752 Ki = 158 nM T67162 D0F4SY 9795739 Ki = 7521 nM T67162 D0HZ2E 5311271 Ki = 1300 nM T67162 D0L3JI 188942 Ki = 2230 nM T67162 D0LI1C 44469321 IC50 > 10000 nM T67162 D0N1HW 5311200 Ki = 448 nM T67162 D0R9HI 11256720 Ki = 997 nM T67162 D0W5EH 6918388 IC50 < 6 nM T67162 D0X2XF 177336 Ki < 1000 nM T67162 D0Y6HW 107930 Ki = 980 nM T67162 D04UXX 3075615 Ki = 5.2 nM T67162 D07YLK 4350931 Ki = 19 nM T67162 D0K5EE 9868452 Ki = 31.62 nM T67162 D0Q3GV 15389743 Ki = 1202.26 nM T67162 D0U0YR 11520239 Ki = 2800 nM T67162 D00KZF 2419 Ki = 14 nM T67162 D00PXQ 60785 Ki = 180 nM T67162 D01DAW 208951 Ki = 0.04 nM T67162 D01PIL 54477 IC50 = 1.202 nM T67162 D01RAE 133079 Ki = 5147 nM T67162 D01WJZ 60820 Ki = 2.2 nM T67162 D01ZSF 24840389 Ki = 630.96 nM T67162 D02FNU 56971 Ki = 110 nM T67162 D02JMI 9888211 Ki = 3.162 nM T67162 D02VUX 11697676 Ki = 0.81 nM T67162 D03TNA 5025739 Ki = 160 nM T67162 D03YPJ 5163 Ki < 10000 nM T67162 D03ZZH 9887537 Ki = 3.981 nM T67162 D06DZI 107780 Ki < 10000 nM T67162 D07ODD 132891 Ki = 158 nM T67162 D08AWI 11430856 Ki > 2000 nM T67162 D09DRG 9952420 IC50 > 10000 nM T67162 D09WHM 208917 Ki = 0.42 nM T67162 D0A3OF 10026300 IC50 = 52 nM T67162 D0B7SP 11292933 Ki = 501.19 nM T67162 D0BN4Y 9797080 Ki > 50000 nM T67162 D0C5PA 183812 EC50 = 1.995 nM T67162 D0EE6L 3038495 Ki = 33.6 nM T67162 D0FH3X 9916104 Ki = 351 nM T67162 D0K9JP 9928332 Ki > 1000 nM T67162 D0L5TJ 10527469 Ki = 19.7 nM T67162 D0M7LV 5761 Ki = 120 nM T67162 D0M9GE 53389 Ki > 10000 nM T67162 D0OS6O 60149 Ki = 0.45 nM T67162 D0OU7P 1242 Ki = 720000 nM T67162 D0P2YS 6603703 Ki = 1550 nM T67162 D0Q2JS 10436045 Ki = 15.85 nM T67162 D0R5GS 55191 Ki = 58 nM T67162 D0T1SF 9909448 Ki = 241 nM T67162 D0TH1Z 57533 Ki = 6.24 nM T67162 D0UZ1I 9841864 Ki = 39.81 nM T67162 D0Y6GJ 176407 EC50 > 100000 nM T67162 D0Y6SN 5311096 Ki = 398.11 nM T67162 D0YP7L 6604889 Ki = 316 nM T67162 D0Z2WQ 57242 EC50 = 2 nM T67162 D0Z4QV 121967 Ki = 1630 nM T67162 D0Z7AW 9820261 Ki > 3310 nM T67162 D0ZG9N 132337 Ki > 10000 nM T67162 C7DT6H 15115517 Ki = 0.3 nM T67162 CY9E4K 15115518 Ki = 0.45 nM T67162 C7ALK2 1240 Ki = 0.5 nM T67162 COJD92 1687 Ki = 1740 nM T67162 CZUI83 2769 IC50 = 227 nM T67162 C0H8GR 3191 IC50 = 61 nM T67162 CT2N1A 4249 Ki = 0.7244 nM T67162 CW56ZA 5290 Ki = 115.5 nM T67162 C54IUQ 5357 Ki = 6.31 nM T67162 C0OCW6 6240 Ki = 3 nM T67162 C5H9CN 9287 Ki > 10000 nM T67162 CVW5J9 10220 Ki = 102 nM T67162 CRD7M3 11492 Ki = 20000 nM T67162 C3A6IG 16103 Ki = 2500 nM T67162 C2JW4U 18367 Ki = 7.586 nM T67162 C8OW9T 18519 Ki = 3400 nM T67162 C9E6DA 21171 Ki = 80.2 nM T67162 C87UJB 21454 Ki > 1300 nM T67162 C17TDE 23269 Ki > 10000 nM T67162 CFGH18 27620 Ki = 49 nM T67162 CT60VY 32224 Ki = 2.5 nM T67162 C5EGZ1 34580 Ki = 1.4 nM T67162 C8Y6DE 37461 IC50 = 0.000000005 nM T67162 CG1A3M 38282 Ki = 9090 nM T67162 CD9E4R 44668 Ki > 1000 nM T67162 CJS51G 52919 Ki = 0.46 nM T67162 CGB1S7 57532 Ki = 0.3388 nM T67162 COI7E6 59227 Ki = 0.06 nM T67162 CBJ5R0 65340 EC50 = 0.631 nM T67162 C97NOS 68634 Ki = 5.5 nM T67162 C6CU1T 70515 Ki > 10000 nM T67162 C5J8VT 86131 Ki = 128 nM T67162 C6MRZ3 91588 Ki = 5000 nM T67162 CK16NU 92716 Ki = 1900 nM T67162 CAL9G2 92910 Ki = 0.04 nM T67162 CZ8P9S 94688 IC50 = 10 nM T67162 CPZ5N6 98358 Ki > 10000 nM T67162 C12BFY 114840 Ki = 3900 nM T67162 C9NJK8 114876 EC50 = 39 nM T67162 CM34NA 119265 Ki = 91.2 nM T67162 CI24CD 120540 Ki = 478 nM T67162 C9VZR2 121852 IC50 = 10 nM T67162 CKP25M 121881 Ki < 10000 nM T67162 CKR4N3 122065 Ki = 32 nM T67162 CN9X8Q 122132 Ki = 340 nM T67162 CDX16S 122167 EC50 = 0.7 nM T67162 C9IBE6 125156 Ki = 1492 nM T67162 C1B4NI 125328 Ki = 640 nM T67162 CG21YH 127262 Ki > 1000 nM T67162 C5SWN1 127698 Ki = 8.4 nM T67162 CI47KZ 127708 Ki = 854 nM T67162 C9BYH2 128032 Ki > 10000 nM T67162 CD2C0M 128054 Ki = 0.14 nM T67162 CZIL53 130844 Ki = 77 nM T67162 C5C2MK 131001 Ki > 3000 nM T67162 C9WG8X 131559 Ki = 1.7 nM T67162 C53TUG 132435 EC50 = 122 nM T67162 CC58NU 132955 EC50 = 1 nM T67162 CS8W1F 133642 EC50 = 7.7 nM T67162 CZL87W 133999 IC50 > 10000 nM T67162 C7I3TL 147514 Ki = 160 nM T67162 C6CW2T 151086 Ki = 338.84 nM T67162 C1ND9W 161665 Ki = 305 nM T67162 C9OD2N 163091 Ki = 8.9 nM T67162 CLK7P3 169713 IC50 > 10000 nM T67162 CF7O0K 171187 Ki = 10 nM T67162 C3Q2NW 173712 Ki = 5.012 nM T67162 CRL1X5 178078 Ki = 0.2 nM T67162 C91DAE 185394 Ki = 26 nM T67162 CVUZ41 185395 Ki = 49 nM T67162 CXS17Y 188442 Ki > 5000 nM T67162 C9XWA6 198914 Ki = 88000 nM T67162 CP2DY7 198967 Ki > 300000 nM T67162 C2INS1 201536 EC50 = 12.59 nM T67162 C16AKU 203697 Ki = 158.49 nM T67162 CVI6X5 213046 Ki = 1.7 nM T67162 C5RC4G 231915 Ki = 217 nM T67162 CYO3R2 300430 Ki > 10000 nM T67162 CHZ1P6 380039 Ki = 71.4 nM T67162 CGZ34T 418856 Ki > 10000 nM T67162 C3HFE4 422923 Ki = 470 nM T67162 CD8Z9H 424430 Ki = 1600 nM T67162 C4O6RK 435595 Ki > 1000 nM T67162 CAH2S5 439654 Ki = 214 nM T67162 CG2JX9 440229 Ki = 41.8 nM T67162 CV6D3N 443374 Ki = 25.12 nM T67162 CFJ3R2 452533 Ki = 130 nM T67162 CHB7D2 453215 IC50 = 3110 nM T67162 C28ARG 511482 Ki = 71 nM T67162 CG59VA 511484 Ki > 300 nM T67162 C17XTV 652557 Ki > 10000 nM T67162 CGIY90 688272 IC50 = 0.00000002 nM T67162 CZN6S9 743974 IC50 > 30199.52 nM T67162 CU8H9L 749986 Ki = 1400 nM T67162 CD7P8Y 763194 Ki > 10000 nM T67162 C6QLR0 763343 Ki > 10000 nM T67162 CLR75J 763625 Ki > 10000 nM T67162 C5SXQ1 763774 Ki > 10000 nM T67162 CW8R4B 778880 Ki > 8300 nM T67162 C9IK2J 792265 Ki = 264 nM T67162 C13TYL 792460 Ki = 162 nM T67162 C4AY9X 792584 Ki = 255 nM T67162 CW0CU9 798232 Ki > 10000 nM T67162 C08WCU 851833 Ki = 137.3 nM T67162 CJ30IQ 1248739 Ki = 19000 nM T67162 CVTP62 1811569 Ki > 10000 nM T67162 C0N4WD 1946142 Ki = 1434 nM T67162 CJI01N 2099556 Ki > 10000 nM T67162 CX85VC 2581635 Ki > 10000 nM T67162 C6N8EF 2812861 Ki = 2190 nM T67162 C3DN1I 2822063 Ki = 598 nM T67162 C1S8CM 2845719 IC50 > 100 nM T67162 CT80MF 3033200 EC50 = 0.3715 nM T67162 C4TB0I 3036864 Ki = 891.25 nM T67162 C64CZV 3038494 Ki = 61 nM T67162 CE4KC8 3038603 Ki = 0.66 nM T67162 C54FEG 3039881 Ki = 2 nM T67162 CT51WS 3045992 EC50 = 0.3 nM T67162 C6Z4QI 3050372 Ki = 119 nM T67162 C5NA6S 3069135 Ki = 37 nM T67162 CS5F1I 3083481 Ki = 1700 nM T67162 CB1FL9 3085297 Ki = 30 nM T67162 CBL51N 3156990 Ki = 1400 nM T67162 C82GMT 3246443 Ki = 49.2 nM T67162 C0U6EW 3504099 Ki = 473 nM T67162 C7YQD3 3519055 Ki = 3683 nM T67162 CCH45N 3626837 IC50 > 1000 nM T67162 C0YXV3 3676358 Ki > 10000 nM T67162 CD76NG 3691783 Ki = 254 nM T67162 CK3W2U 3716121 Ki = 24 nM T67162 C9J5YC 3746693 Ki = 240 nM T67162 CI50PT 4064333 Ki > 1000 nM T67162 CO0FZ1 4064342 Ki = 86 nM T67162 CY7PH0 4302960 Ki = 39.81 nM T67162 CR1L9E 4466165 Ki = 12.02 nM T67162 CRUB15 4723431 Ki = 676 nM T67162 CS6P5D 4797946 EC50 = 763 nM T67162 CWB9I2 4987774 Ki = 17.3 nM T67162 CW2C1I 5009938 Ki > 10000 nM T67162 C6FM8G 5029739 Ki > 1700 nM T67162 C6AQP8 5249952 Ki = 943 nM T67162 C9AZ2I 5249956 Ki = 8.47 nM T67162 CMX45W 5311346 Ki = 20.5 nM T67162 C9FYP1 5312124 Ki = 501.19 nM T67162 CU3L6O 6142670 Ki = 1072 nM T67162 CW34VC 6160690 Ki > 1000 nM T67162 C8R4JX 6305587 Ki = 6.6 nM T67162 CXP45C 6430941 EC50 > 10000 nM T67162 CHO8D2 6453963 EC50 = 56000 nM T67162 C6L9DT 6466372 EC50 = 2092 nM T67162 CWNZ35 6469693 Ki = 110 nM T67162 CJTQ40 6469918 Ki = 15000 nM T67162 CVBX47 6603800 Ki = 20 nM T67162 CIZ7U3 6603820 Ki = 58 nM T67162 CXZ53N 6603866 Ki = 90 nM T67162 CKP56W 6603867 Ki = 0.5 nM T67162 CSM9T8 6603950 Ki = 7.3 nM T67162 C6I3MZ 6603954 Ki = 2.1 nM T67162 C3A1FO 6604789 Ki < 100000 nM T67162 CIB7K3 6604864 Ki > 10000 nM T67162 C5WH0F 6604868 Ki > 5000 nM T67162 CC6SM3 6618861 Ki = 25.8 nM T67162 C8QM7B 6852376 Ki = 4670 nM T67162 C0QCK1 6918455 Ki = 2511.89 nM T67162 CW0ZE5 6918542 Ki = 210 nM T67162 CC5PQ0 6918601 Ki > 1700 nM T67162 C1WXY3 6918603 Ki < 10000 nM T67162 CD0Z4I 6918648 Ki = 794.33 nM T67162 C1R4IO 6937303 Ki = 1060 nM T67162 C6MR7E 8529065 Ki > 300 nM T67162 C3NK0H 8690650 Ki > 300 nM T67162 C9R7NM 9104271 IC50 = 690 nM T67162 C8ZD1I 9129986 Ki = 673 nM T67162 C07UXF 9268266 IC50 = 15700 nM T67162 CVF3N1 9475051 IC50 > 50000 nM T67162 C1MHE9 9549058 IC50 = 2590 nM T67162 CO40CQ 9794644 Ki = 641 nM T67162 C5FUS9 9795741 Ki > 217 nM T67162 CCM0S1 9796255 Ki = 13 nM T67162 CUD06Z 9796627 Ki > 2200 nM T67162 CO5VP3 9796958 Ki = 4020 nM T67162 CC5Z9T 9797161 IC50 = 45 nM T67162 CY6WB3 9797495 Ki = 5700 nM T67162 CLUT03 9799123 Ki = 140 nM T67162 CEG5Z6 9799491 Ki > 1000 nM T67162 CZI29U 9799781 Ki = 209 nM T67162 CKM1U6 9800010 Ki = 15.9 nM T67162 C0TX4L 9800145 Ki = 0.4 nM T67162 CI4S6Y 9800164 Ki = 92 nM T67162 CFR7L3 9801098 Ki = 3027 nM T67162 CX7I8J 9802187 Ki = 4.7 nM T67162 CE0DI5 9804612 Ki < 10000 nM T67162 CNX4F0 9805456 Ki < 3162.28 nM T67162 C59RXH 9816005 Ki = 119 nM T67162 CV5L1J 9817253 Ki = 3.9 nM T67162 CJ78ZE 9817612 Ki > 10000 nM T67162 C6V0MU 9817774 Ki = 3 nM T67162 CWOS30 9817810 Ki > 1700 nM T67162 C9MH4N 9818423 Ki = 302 nM T67162 CHQI10 9818448 Ki = 62.7 nM T67162 C8NIP0 9819042 Ki = 39 nM T67162 CEW91X 9819119 IC50 > 10000 nM T67162 C2V7HU 9819770 Ki = 1842 nM T67162 C0XE2V 9820048 Ki = 1373 nM T67162 CQE93H 9820085 Ki > 5000 nM T67162 C3JBY9 9820304 Ki = 93 nM T67162 CR17LP 9820313 Ki = 132 nM T67162 CVMR82 9820327 Ki = 31.62 nM T67162 CO9VA3 9820671 IC50 > 1000 nM T67162 C1HNW6 9820680 Ki = 32.4 nM T67162 C9D4HQ 9821010 Ki = 1880 nM T67162 COJ3V6 9821803 Ki = 2600 nM T67162 CL38GM 9826580 Ki = 24.8 nM T67162 C0AU9L 9826801 Ki = 140 nM T67162 C8LP9E 9827991 Ki = 76.4 nM T67162 C8EC9B 9828617 Ki = 398 nM T67162 C2F5OX 9828632 Ki > 10000 nM T67162 COG0R8 9836900 Ki = 129 nM T67162 C2MN0P 9837094 Ki = 1281 nM T67162 CO7HQ5 9837137 Ki = 4166 nM T67162 CV2A3K 9838959 Ki > 1000 nM T67162 CBN06W 9839050 Ki = 61 nM T67162 C4BPW7 9839426 Ki = 5.2 nM T67162 C5EDO7 9839491 Ki = 3506 nM T67162 CHSR07 9840044 Ki = 2189 nM T67162 C8XER9 9840365 Ki = 244 nM T67162 C1U6ZX 9840672 Ki = 1.75 nM T67162 C7O0TI 9841203 Ki = 12.59 nM T67162 CS2M1N 9841398 Ki = 710 nM T67162 CF87HQ 9841608 Ki > 5000 nM T67162 CR31XS 9843031 Ki = 2629 nM T67162 CKZ0X3 9843032 Ki = 4375 nM T67162 C2RQ5H 9843062 Ki = 0.19 nM T67162 CN09KS 9843137 Ki = 2610 nM T67162 C8BW3K 9843389 Ki = 69 nM T67162 C80IET 9843967 IC50 > 10000 nM T67162 C02XRE 9844106 Ki = 20 nM T67162 C5MHS3 9847013 Ki = 62 nM T67162 C4B6JU 9847363 Ki = 0.6 nM T67162 CNB65K 9848303 Ki = 310 nM T67162 CJ8LT7 9848518 IC50 > 10000 nM T67162 C21SZB 9848933 Ki > 1000 nM T67162 C7S1YV 9849443 Ki = 1000 nM T67162 C8HMK2 9858274 Ki = 935 nM T67162 C07TSW 9859120 Ki = 265 nM T67162 C7EZ2L 9859861 Ki = 2066 nM T67162 CT78EC 9860183 Ki = 176 nM T67162 C4GT3Z 9861459 Ki = 3 nM T67162 CD12MS 9861786 Ki = 2.6 nM T67162 CNCK78 9862256 Ki = 1600 nM T67162 C4YA9P 9863108 Ki = 19.95 nM T67162 C8M5XK 9863333 Ki = 1431 nM T67162 C0Q6AD 9863611 Ki = 158.49 nM T67162 CKF2T8 9864325 Ki = 140 nM T67162 CBW2I4 9864749 Ki > 10000 nM T67162 CTY02P 9865254 Ki = 2200 nM T67162 CI30XR 9865463 Ki = 2.3 nM T67162 C1SM8I 9865490 Ki = 271 nM T67162 CR06ME 9865584 Ki = 38 nM T67162 C5WYN4 9865858 Ki = 13.2 nM T67162 CWN76A 9865920 Ki = 607 nM T67162 C7EX8O 9867004 Ki = 187 nM T67162 C4IZ3J 9867233 Ki = 1178 nM T67162 CB1F0C 9867475 Ki = 750 nM T67162 CJAU58 9868502 Ki = 39.81 nM T67162 C7AB8O 9870053 Ki < 1000 nM T67162 CT2C6K 9870702 IC50 > 10000 nM T67162 C2ELZ9 9881053 IC50 = 3400 nM T67162 C9NF3D 9881600 Ki = 450 nM T67162 CL0F2R 9881980 Ki = 398.11 nM T67162 C7KP4G 9882069 Ki > 10000 nM T67162 C8L6GE 9882257 Ki = 11 nM T67162 C10MKO 9882537 Ki > 1000 nM T67162 CX8M6A 9883221 Ki = 1168 nM T67162 COI69G 9883554 Ki = 3019.95 nM T67162 CW97YN 9883587 Ki = 436 nM T67162 C3DB5H 9884781 Ki = 738 nM T67162 CTAC24 9885114 Ki = 413 nM T67162 COT4C7 9885219 Ki = 195 nM T67162 CZ8C7G 9885279 Ki > 1500 nM T67162 C64EOU 9885465 Ki = 1400 nM T67162 CC16TR 9885927 Ki = 11.3 nM T67162 C1FG7S 9886340 Ki = 4623 nM T67162 CALV92 9886609 EC50 = 2.8 nM T67162 CH84KI 9887091 Ki = 117 nM T67162 CYRS07 9887092 Ki > 1000 nM T67162 CQ03IA 9887463 Ki = 2.5 nM T67162 CJW1P5 9888494 Ki = 234.42 nM T67162 C9GB2M 9888555 Ki = 25 nM T67162 CDLB96 9889149 IC50 = 140 nM T67162 C6N8UE 9889681 Ki < 5011.87 nM T67162 CN6L8E 9889735 Ki = 398.11 nM T67162 C2XAH9 9889736 Ki = 630.96 nM T67162 CM52WU 9890119 Ki < 5011.87 nM T67162 CEG1K5 9891002 Ki < 3981.07 nM T67162 C7QMK5 9891617 Ki < 6309.57 nM T67162 CEL29O 9891618 Ki < 7943.28 nM T67162 C6WY0D 9891901 Ki = 54.7 nM T67162 C3J8GU 9892409 Ki = 398.11 nM T67162 CAM25C 9894665 Ki = 23 nM T67162 CZ7D4L 9901646 Ki = 515 nM T67162 CBI9C5 9901894 IC50 = 246 nM T67162 CR8GO9 9902381 Ki = 493 nM T67162 C1U3EY 9902382 Ki = 2980 nM T67162 C5TA6D 9903398 Ki > 1000 nM T67162 CUPI23 9903623 Ki = 3090.3 nM T67162 C6RGI9 9904074 Ki = 27 nM T67162 CFI97S 9904205 IC50 = 870.96 nM T67162 CNO38Q 9905222 Ki > 10000 nM T67162 CUN81Q 9905249 Ki > 1500 nM T67162 CYWQ50 9906447 Ki > 10000 nM T67162 CD3F4N 9906454 Ki > 5000 nM T67162 C6CZ3G 9906777 IC50 > 10000 nM T67162 C7XS1O 9906895 Ki = 980 nM T67162 C7JFZ5 9906978 Ki = 33 nM T67162 CDE29K 9907381 Ki > 10000 nM T67162 CY51ZT 9907436 Ki = 0.003 nM T67162 C07SWP 9907461 Ki > 5000 nM T67162 CT96CK 9908071 Ki = 7367 nM T67162 C6YKE0 9908125 Ki = 480 nM T67162 C2Z9BL 9908431 Ki > 1500 nM T67162 CY2I0L 9908478 Ki = 120 nM T67162 C7SMT0 9908904 IC50 > 1000 nM T67162 CMZ58L 9909055 Ki > 10000 nM T67162 CYZ5N4 9909089 Ki = 316.23 nM T67162 C5AHG4 9909521 Ki = 55 nM T67162 C3NOI2 9909614 Ki = 406 nM T67162 CO7BK6 9909648 Ki = 199 nM T67162 C4L2CV 9911120 IC50 = 1096.48 nM T67162 CXV7O3 9912796 Ki = 398.11 nM T67162 C78MDV 9913554 Ki = 1584.89 nM T67162 CB6J3C 9913988 Ki = 2.7 nM T67162 C8LJ9H 9914930 Ki = 630.96 nM T67162 CE7UF1 9925530 Ki = 758.58 nM T67162 CJL38X 9925730 Ki = 15.2 nM T67162 CZ4WE9 9927411 Ki = 2235 nM T67162 C4UYZ7 9927441 Ki = 62 nM T67162 CB12RM 9929629 Ki > 1000 nM T67162 C2H8FQ 9930722 Ki > 1000 nM T67162 CN4HQ8 9930934 Ki = 1096 nM T67162 C1C5KY 9931327 Ki = 700 nM T67162 CM3X7Y 9931571 Ki > 1000 nM T67162 CN3OW2 9932051 Ki = 1.7 nM T67162 CP45YZ 9932385 Ki = 1000 nM T67162 CAQ52T 9932698 Ki = 37 nM T67162 CUHL40 9933550 Ki = 3162.28 nM T67162 CYVZ47 9934284 Ki = 1995.26 nM T67162 CWO45F 9935387 Ki = 1995.26 nM T67162 C8BX2L 9945233 Ki > 10000 nM T67162 C1ES5F 9946469 Ki = 346 nM T67162 CZPM75 9948461 Ki = 519 nM T67162 CU2JM9 9948584 Ki = 5 nM T67162 C8T1HO 9948670 Ki = 28 nM T67162 C9EUM1 9948965 Ki = 364 nM T67162 CO2QA0 9949442 Ki = 140 nM T67162 CA07XW 9949531 Ki = 6.5 nM T67162 CIFG92 9949601 Ki > 5000 nM T67162 C02IMR 9949655 IC50 = 300 nM T67162 CXEZ63 9950165 Ki = 56 nM T67162 CQ04ZS 9950396 Ki > 300000 nM T67162 CS95KP 9950913 Ki > 1000 nM T67162 C1K8WB 9951233 Ki = 133 nM T67162 CZ6D4W 9951735 Ki = 8.6 nM T67162 C8DQ6P 9952003 Ki = 9 nM T67162 C92UQN 9952218 Ki > 1000 nM T67162 CHU17Z 9952528 Ki = 100 nM T67162 CKF9X1 9953268 Ki = 1000 nM T67162 CEL95F 9953774 Ki = 630.96 nM T67162 CK8NR2 9954121 Ki < 10000 nM T67162 CWSE34 9954899 IC50 = 140 nM T67162 CC18QK 9955015 Ki > 10000 nM T67162 CU2C3V 9955072 Ki = 1.5 nM T67162 CFR41N 9957068 Ki = 501.19 nM T67162 CZB52R 9967004 Ki = 2200 nM T67162 CGP43F 9967140 IC50 = 5 nM T67162 CIW4R8 9968343 Ki = 2340 nM T67162 CTNH36 9972630 Ki = 590 nM T67162 C25BNI 9975434 Ki = 59.2 nM T67162 CC1ZL3 9975465 Ki = 897 nM T67162 CKU4N1 9976024 Ki = 16 nM T67162 CXT1W6 9977478 Ki = 0.65 nM T67162 CMYN90 9977532 Ki = 2 nM T67162 CU6T9Q 9977907 Ki = 83.18 nM T67162 CFN50J 9978683 Ki = 334 nM T67162 CC6M7Z 9980998 Ki = 44.8 nM T67162 CRI0K3 9981035 Ki = 96 nM T67162 CC05RX 9982218 Ki = 63 nM T67162 C4G1IX 9982854 Ki = 95.5 nM T67162 CT7G0Y 9983212 Ki = 216 nM T67162 C56XEZ 9983667 Ki = 936 nM T67162 CB8NT0 9991216 Ki > 217 nM T67162 C9BM2I 9991512 Ki = 145 nM T67162 CGWR69 9992102 Ki = 87 nM T67162 CXQ5O2 9992189 Ki = 5 nM T67162 CP41ZO 9992499 Ki = 264 nM T67162 CK54BS 9992778 Ki = 327 nM T67162 C8K6NO 9992903 Ki = 1202 nM T67162 C7FVY2 9994243 Ki = 40 nM T67162 CB2EP7 9995264 Ki = 774 nM T67162 CUS7W9 9995379 Ki = 8 nM T67162 CP31VK 9995904 Ki = 290 nM T67162 C5AO4D 9998085 Ki = 344 nM T67162 CV4BN3 9999267 Ki = 9.7 nM T67162 CE17DV 10000260 IC50 = 1.413 nM T67162 C7NC3D 10000302 Ki = 3950 nM T67162 C6FA2J 10001207 Ki = 1500 nM T67162 C17ZTJ 10001256 Ki = 2.9 nM T67162 C0DIO1 10001810 Ki = 273 nM T67162 C1NQC9 10003809 Ki = 67.61 nM T67162 CQL12P 10004545 Ki = 3160 nM T67162 CL9QS0 10004950 IC50 = 2120 nM T67162 C27WPA 10007017 Ki = 2290.87 nM T67162 C6TJI2 10009952 Ki = 1495 nM T67162 CSJQ56 10013665 Ki > 217 nM T67162 CM26VE 10014056 Ki = 75 nM T67162 CO39AR 10014057 Ki = 0.3 nM T67162 CUX43N 10014136 Ki < 50 nM T67162 CIX9P8 10014484 EC50 > 10000 nM T67162 CUIQ94 10014924 Ki = 41 nM T67162 C5MUC9 10015045 Ki = 58.5 nM T67162 CS40QN 10015688 Ki = 1300 nM T67162 C5ZJ4W 10015731 Ki = 1.14 nM T67162 C61KDJ 10015860 Ki = 2500 nM T67162 CFM38B 10017758 Ki = 44 nM T67162 CFP13M 10018300 Ki = 91 nM T67162 CTK42D 10018480 Ki = 83 nM T67162 C9LC6Z 10020651 Ki = 3346 nM T67162 CAY37B 10020914 Ki = 0.05 nM T67162 C94EDH 10021099 Ki = 515 nM T67162 C1VDL8 10021193 Ki = 600 nM T67162 CXBN42 10021692 Ki = 0.097 nM T67162 CS83XQ 10022628 Ki = 25 nM T67162 C5X1KG 10022781 Ki = 45.71 nM T67162 CE9NR0 10024832 Ki = 1.259 nM T67162 C8ECG9 10025039 EC50 = 240 nM T67162 CRTY53 10025040 EC50 > 1000 nM T67162 C7MVE2 10027629 Ki = 610 nM T67162 CUC01W 10036468 EC50 > 10000 nM T67162 CM0Z7A 10036887 Ki = 917 nM T67162 C9LF0P 10037311 Ki > 217 nM T67162 CPXC69 10037436 Ki = 50 nM T67162 C3MK8V 10039198 Ki = 16 nM T67162 CGTA58 10040546 Ki = 730 nM T67162 C1MJV4 10041417 Ki = 0.76 nM T67162 CM3L5T 10041887 Ki = 1137 nM T67162 C3RPO9 10042466 Ki = 37 nM T67162 C2C1XS 10042602 Ki = 51.29 nM T67162 CN1M6G 10042972 Ki = 2780 nM T67162 CIBU84 10043468 Ki = 1969 nM T67162 C0HVU6 10044835 Ki = 2550 nM T67162 CJ3V7G 10045023 Ki = 410 nM T67162 CFXD46 10045525 Ki = 21 nM T67162 CA42DO 10047196 Ki > 5000 nM T67162 CK5GJ9 10047648 EC50 = 10.4 nM T67162 CYN90C 10047649 EC50 > 1000 nM T67162 C2JZL1 10048222 IC50 > 1000 nM T67162 C8WPO6 10049549 Ki = 7585.78 nM T67162 CX27EK 10049758 IC50 = 23 nM T67162 CRZ48G 10050500 Ki = 1584.89 nM T67162 CWGQ38 10052229 Ki = 630.96 nM T67162 CNU12A 10052433 Ki = 25.12 nM T67162 C4GHO2 10053476 Ki = 48 nM T67162 CLNY93 10058787 Ki = 3.8 nM T67162 CFXB93 10059206 Ki = 12 nM T67162 C2G9HJ 10060349 Ki > 217 nM T67162 C5ZLK0 10060449 Ki > 217 nM T67162 CL23OT 10060538 Ki = 6.24 nM T67162 C74CWJ 10061323 Ki = 79.2 nM T67162 C0KWB6 10062885 Ki = 7.1 nM T67162 C6Y3NO 10063875 Ki = 9.3 nM T67162 C9W8ZV 10063953 Ki = 65.6 nM T67162 CUW74G 10064052 Ki = 241 nM T67162 CR68SH 10064053 Ki = 233 nM T67162 CQ2CS1 10064981 Ki > 10000 nM T67162 C4PCO3 10065083 Ki = 98 nM T67162 CT2OG9 10065188 Ki = 177.83 nM T67162 CYX3E7 10065496 Ki = 1272 nM T67162 COZU58 10066419 Ki = 540 nM T67162 C3TJ0U 10066604 Ki = 12.6 nM T67162 C0ISR6 10067170 Ki = 389 nM T67162 C8Z6MA 10067306 IC50 < 5000 nM T67162 CO69FB 10069973 Ki = 78.1 nM T67162 C4LQY1 10071413 Ki = 141.25 nM T67162 C2JFB1 10072280 Ki = 8.8 nM T67162 C5HJ1G 10073022 Ki = 81.3 nM T67162 C03KWH 10073194 Ki = 119 nM T67162 C0V5ZR 10074155 Ki = 8 nM T67162 C75OQF 10075078 Ki = 794.33 nM T67162 CKA5F4 10084076 Ki = 2250 nM T67162 CJ16VZ 10084583 Ki = 35 nM T67162 CW7MA3 10084845 Ki > 50000 nM T67162 CB8K0C 10086123 Ki = 250 nM T67162 CX6L2Q 10086348 EC50 = 1.3 nM T67162 C03CYX 10086395 Ki = 29 nM T67162 CV04JN 10087023 IC50 > 1000 nM T67162 CGW9L7 10088259 Ki = 380.19 nM T67162 C2M6UR 10088426 Ki = 50 nM T67162 CQVJ58 10088453 Ki = 5.37 nM T67162 C6BDZ3 10089203 Ki = 188 nM T67162 CIMQ96 10090127 Ki = 219 nM T67162 CVK93I 10090424 Ki = 16.22 nM T67162 C63FME 10090486 Ki = 724.44 nM T67162 C0XB2Y 10090714 Ki > 5000 nM T67162 CR3D5E 10091430 IC50 = 67.61 nM T67162 C7O8VH 10092041 IC50 = 150 nM T67162 C8NQ3I 10092649 IC50 = 5100 nM T67162 CJXQ40 10092819 Ki = 84 nM T67162 CA3LE2 10098342 Ki = 10000 nM T67162 CD3Y1G 10105186 Ki = 106 nM T67162 CH5WC1 10105311 Ki = 0.5 nM T67162 C7NK1P 10105359 Ki = 272 nM T67162 C0XO1J 10105844 Ki = 6.7 nM T67162 C5PJ3N 10107367 Ki = 1862.09 nM T67162 C54EYD 10108561 IC50 = 1905.46 nM T67162 CKCI50 10110263 Ki = 2530 nM T67162 C7QEX4 10114519 EC50 = 6.3 nM T67162 C0HAD8 10115074 Ki = 220 nM T67162 CF1LH5 10130293 Ki > 10000 nM T67162 CVD86L 10130933 Ki = 27 nM T67162 CL7N8S 10131111 Ki = 402 nM T67162 COXA05 10133031 Ki = 206 nM T67162 CS1B5X 10137322 Ki = 610 nM T67162 CWT32F 10137747 Ki = 313 nM T67162 C8X4BP 10137748 Ki = 952 nM T67162 C5JZ9P 10157556 Ki = 62 nM T67162 CR62CZ 10158455 Ki = 139 nM T67162 C1DQ8L 10161526 Ki = 620 nM T67162 CBW5L2 10169960 Ki > 1000 nM T67162 CP6Q1W 10173403 Ki = 158.49 nM T67162 CZ3RL4 10176243 Ki = 11400 nM T67162 CB30TC 10176799 Ki = 462 nM T67162 C8M2KL 10178704 EC50 = 12.2 nM T67162 CUN52S 10183297 Ki = 470 nM T67162 C2ZC0Q 10183626 Ki = 1461 nM T67162 CZ97UO 10184153 Ki = 491 nM T67162 C7Y3JR 10200368 Ki = 245 nM T67162 CZKG96 10200496 Ki = 0.55 nM T67162 CFJY39 10216820 Ki = 31.62 nM T67162 CV1B7C 10217687 Ki = 3.981 nM T67162 CMJ2W9 10220333 Ki = 111 nM T67162 CWR4J6 10220541 Ki = 1350 nM T67162 CC38UK 10221294 EC50 > 1000 nM T67162 CY2S4Z 10224165 Ki = 201 nM T67162 CGJ5Q9 10225942 Ki = 486 nM T67162 C47KBM 10228202 Ki = 8.78 nM T67162 CS3X6I 10229397 Ki = 2618 nM T67162 CYAV42 10236153 Ki = 5000 nM T67162 CO64WJ 10236758 Ki = 676.08 nM T67162 C8B4SV 10241065 Ki = 53800 nM T67162 COZ2S7 10242548 Ki = 380 nM T67162 C7LY2Z 10242819 Ki > 217 nM T67162 C5PDQ8 10242850 Ki > 217 nM T67162 CYCQ58 10245409 Ki = 200 nM T67162 CVF1E5 10246054 IC50 = 446.68 nM T67162 CYT27X 10247457 Ki = 3 nM T67162 CC3XF5 10247561 Ki = 66000 nM T67162 CG2B7I 10247701 Ki = 1.66 nM T67162 CFCP96 10247720 Ki = 10000 nM T67162 CY82IS 10248715 Ki > 1900 nM T67162 C6SB5G 10249134 Ki = 300 nM T67162 C4Q2SH 10249573 Ki = 630.96 nM T67162 CWD35Q 10249755 Ki = 7943.28 nM T67162 C0XJ2W 10250895 Ki = 11.75 nM T67162 CC1PJ7 10251080 Ki = 194 nM T67162 C2UNO6 10251160 Ki = 73 nM T67162 C3QGA5 10251795 IC50 = 2060 nM T67162 CSPF93 10252272 Ki = 398.11 nM T67162 C6SNB5 10252580 Ki = 447 nM T67162 C7NO2S 10253333 Ki = 307 nM T67162 C9XTQ2 10253970 Ki = 7.4 nM T67162 COB28U 10254390 Ki = 373 nM T67162 CMRA02 10257042 Ki = 1258.93 nM T67162 C4TK2U 10263215 Ki > 10000 nM T67162 C1FTS4 10263410 Ki > 217 nM T67162 C5RF0W 10264090 Ki > 217 nM T67162 CXM2I0 10264172 Ki > 10000 nM T67162 CE9Y8J 10276451 Ki = 42.5 nM T67162 C9MPY2 10300403 Ki = 1522 nM T67162 C0L8VZ 10301202 Ki = 3828 nM T67162 C36PLT 10313891 Ki = 1000 nM T67162 CU3AC0 10314788 Ki = 600 nM T67162 CJ3Q1T 10314824 Ki = 19000 nM T67162 C5R8TC 10315310 Ki = 228 nM T67162 C5XB6Y 10315866 Ki > 217 nM T67162 CZM6T1 10316192 Ki > 10000 nM T67162 CA3E4W 10316297 Ki = 23.99 nM T67162 CHYJ47 10317514 Ki = 10.8 nM T67162 CB8O9X 10318141 Ki = 3700 nM T67162 CE6V0B 10330427 Ki > 217 nM T67162 C57PKI 10330528 Ki > 217 nM T67162 CE6IP1 10333670 Ki = 54.6 nM T67162 CK5EP8 10333837 Ki = 248 nM T67162 CRQN68 10333842 Ki = 12.7 nM T67162 C6WEU2 10334422 Ki = 22 nM T67162 CHJ4W9 10335148 Ki = 21 nM T67162 C70MLB 10337045 Ki = 1417 nM T67162 C3E5CB 10337773 Ki < 100000 nM T67162 CR3J9S 10338282 Ki = 151.36 nM T67162 CUY3O1 10340117 Ki = 1.8 nM T67162 CNAV40 10340492 Ki = 5.92 nM T67162 C9IAV3 10346043 Ki > 10000 nM T67162 CBAZ60 10353207 Ki > 217 nM T67162 CXO0J4 10353777 Ki = 25 nM T67162 COT48Q 10353846 Ki = 93 nM T67162 CN8JF4 10354398 Ki > 217 nM T67162 C7DQA1 10354437 Ki = 8.5 nM T67162 CUYR47 10355219 Ki = 464 nM T67162 CK7E9M 10355252 Ki = 1330 nM T67162 C0H3VS 10355305 Ki > 217 nM T67162 CXO8I7 10355406 Ki = 45.6 nM T67162 CPK71L 10356389 Ki = 170 nM T67162 CYP68J 10356955 Ki = 82 nM T67162 C4A0PF 10357628 Ki = 61 nM T67162 C1RX9F 10357631 EC50 = 0.5 nM T67162 C1NTD8 10359539 Ki = 29000 nM T67162 CDCX49 10359736 Ki = 2511.89 nM T67162 CXAK13 10359942 Ki > 1600 nM T67162 C32KOP 10360923 Ki > 1700 nM T67162 CD4H6R 10361512 Ki = 58000 nM T67162 C8LT7J 10363821 Ki = 9943 nM T67162 C2A5PV 10364677 Ki = 25.2 nM T67162 CM7L5C 10367367 Ki = 15 nM T67162 CJ6L9D 10368423 Ki = 146 nM T67162 CQEJ41 10368773 Ki = 501.19 nM T67162 C9LWG3 10369004 IC50 = 43 nM T67162 C2X9PQ 10369220 Ki = 168 nM T67162 CH1IY6 10375676 Ki = 0.5 nM T67162 C2OWC5 10377224 Ki = 75 nM T67162 CD9OQ2 10377227 Ki > 217 nM T67162 CIX51R 10378194 Ki = 580 nM T67162 C0O9UQ 10378785 Ki = 265 nM T67162 CA7IM5 10379532 Ki = 71 nM T67162 CD63EZ 10379766 Ki = 420 nM T67162 CL48ZG 10380129 Ki > 217 nM T67162 CR3KU9 10380133 IC50 < 5000 nM T67162 CDAC63 10381889 IC50 = 8.71 nM T67162 CJ01BF 10382430 Ki > 217 nM T67162 C7G9TF 10382446 Ki = 62 nM T67162 C6DFI4 10382581 Ki = 835 nM T67162 CMZA83 10383646 Ki = 355 nM T67162 CCZ74R 10384372 Ki = 125 nM T67162 CEX1T3 10384736 Ki > 217 nM T67162 CER30L 10384998 Ki = 10.8 nM T67162 C69KIB 10385855 IC50 > 10000 nM T67162 CX32VU 10385897 Ki = 124 nM T67162 CLY48W 10385977 IC50 = 20 nM T67162 C7J2TY 10389636 Ki = 199.53 nM T67162 CQ90WG 10390058 Ki = 602 nM T67162 CT3DJ5 10391240 Ki > 217 nM T67162 C4DZ0M 10392655 Ki = 58.8 nM T67162 C4UG3B 10395316 Ki = 343 nM T67162 CD5H6P 10397550 Ki > 217 nM T67162 C64HBT 10398936 Ki = 235 nM T67162 C6J2ZL 10402378 Ki = 158 nM T67162 CIF2V7 10402380 Ki = 179 nM T67162 C8WK6Q 10402381 Ki = 192 nM T67162 CJNR48 10403092 Ki = 524 nM T67162 CT07SM 10403435 Ki = 110 nM T67162 CX2Y7J 10403608 Ki = 75 nM T67162 C4OF7Y 10404663 Ki = 30 nM T67162 CS3OC4 10405678 Ki > 217 nM T67162 C94PNM 10406796 Ki = 467 nM T67162 CM50VF 10406989 Ki = 10.8 nM T67162 C04WGF 10407367 IC50 < 5000 nM T67162 C0HSY3 10409174 Ki = 436.52 nM T67162 C8S3XE 10409556 IC50 = 29.51 nM T67162 CC5A2I 10411237 Ki > 23890 nM T67162 CH5M7W 10413085 Ki = 109.65 nM T67162 C4TPN1 10413595 Ki = 2511.89 nM T67162 CS6W9C 10414769 Ki = 251.19 nM T67162 C60ICT 10420915 Ki > 217 nM T67162 C0HM5D 10421583 Ki = 527 nM T67162 CCM6Y7 10421679 Ki = 20 nM T67162 CX1FR6 10423970 Ki = 1079 nM T67162 CGTF70 10424172 Ki = 89 nM T67162 C2SLJ9 10424961 Ki = 680 nM T67162 CZ5HC6 10425024 EC50 = 0.5 nM T67162 CO76HW 10425969 Ki = 975 nM T67162 CEKH47 10426373 Ki = 554 nM T67162 CA3PI9 10427977 Ki = 3700 nM T67162 CG6S8W 10428643 Ki > 10000 nM T67162 C4YBI9 10428654 Ki > 217 nM T67162 CTG0F9 10429067 Ki = 1210 nM T67162 CG0QM1 10429420 Ki = 2192 nM T67162 C1A8XG 10430305 Ki = 577 nM T67162 CR4LS0 10430623 Ki > 5000 nM T67162 CA1FD2 10430685 Ki = 246 nM T67162 CD86MZ 10430816 Ki = 77 nM T67162 CL0ZB2 10430935 Ki = 228 nM T67162 C0XZB9 10432760 Ki > 100 nM T67162 C8ZA3G 10432808 Ki = 28 nM T67162 CD7U5I 10433930 Ki > 10000 nM T67162 C9A4MJ 10436285 Ki = 19.4 nM T67162 C4UN0A 10436653 Ki = 39 nM T67162 C8KD1B 10438027 Ki = 430 nM T67162 C8MF4H 10438351 Ki = 398.11 nM T67162 C9WB1M 10444260 EC50 > 10000 nM T67162 C1CO4G 10447709 Ki = 389.05 nM T67162 CPN63D 10449136 Ki = 520 nM T67162 CI0N2R 10449738 Ki = 61 nM T67162 CL8HQ6 10450082 IC50 = 9800 nM T67162 C47IOH 10450375 Ki = 1.3 nM T67162 CS1LF0 10450580 Ki > 217 nM T67162 CO7IV6 10450593 Ki = 370 nM T67162 C2G0AH 10450758 Ki = 1100 nM T67162 CVPK09 10450880 Ki > 5800 nM T67162 C1SZU3 10450892 Ki = 299 nM T67162 C9WS1O 10451844 Ki = 3.6 nM T67162 C4LJW3 10452020 Ki = 350 nM T67162 CW0ND4 10454026 Ki = 37.4 nM T67162 CATL09 10455444 Ki = 5 nM T67162 CUB9J6 10456040 Ki = 8.8 nM T67162 C05PSB 10456166 Ki = 103 nM T67162 CK15JL 10456628 Ki = 196 nM T67162 C38VGA 10457264 IC50 = 1500 nM T67162 CWE8U9 10457321 Ki = 1892 nM T67162 CN6CD4 10457955 Ki = 356 nM T67162 CAM7K8 10458892 Ki = 2200 nM T67162 CP17RZ 10466368 Ki = 4.1 nM T67162 C1YS3M 10466454 Ki = 218 nM T67162 CN41CS 10466682 EC50 > 10000 nM T67162 C8RQZ4 10466922 Ki = 69 nM T67162 CZ8X1Q 10466923 Ki = 98 nM T67162 CL6FY4 10466962 Ki = 18 nM T67162 CM23NE 10467118 Ki > 217 nM T67162 CK57FH 10469437 Ki = 230 nM T67162 CV9N7G 10470579 Ki = 67 nM T67162 COV85C 10472143 Ki = 110 nM T67162 C5LBS7 10472158 IC50 < 5000 nM T67162 CUW3M2 10473658 Ki = 269.15 nM T67162 C7HI4X 10474613 Ki = 1438 nM T67162 CPI5M7 10476504 Ki = 99 nM T67162 CI58CV 10476586 Ki = 3500 nM T67162 CE79QV 10477871 Ki = 158.49 nM T67162 CEF2O6 10478367 Ki > 10000 nM T67162 CFLZ47 10479188 Ki = 245 nM T67162 CJI15O 10479214 Ki = 179 nM T67162 CCT42I 10479465 Ki = 27.4 nM T67162 CEP10Q 10479822 Ki = 338.84 nM T67162 CFD83Z 10490043 Ki > 1000 nM T67162 CD3A2O 10492351 Ki > 1600 nM T67162 C2WNH9 10494394 Ki = 292 nM T67162 C4JWB8 10494689 Ki = 77 nM T67162 CB52TQ 10495305 Ki > 1600 nM T67162 CPG8U3 10495787 Ki = 1600 nM T67162 CP51BI 10495881 Ki = 296 nM T67162 CI6PN3 10495891 Ki = 24.5 nM T67162 CQB58X 10496095 IC50 = 752 nM T67162 CV4GF9 10496727 Ki = 582 nM T67162 CG7Y1H 10497177 Ki = 160 nM T67162 C3ZW8P 10497179 Ki = 65 nM T67162 C7VC6L 10497193 Ki = 120 nM T67162 CQ72YM 10497674 IC50 = 13 nM T67162 CX1UD7 10498094 Ki = 950 nM T67162 CHUF43 10498196 Ki = 1130 nM T67162 CRUT74 10498972 Ki = 5730 nM T67162 C9M3FN 10499950 Ki = 7.4 nM T67162 C31HYJ 10501113 IC50 = 250 nM T67162 C71MTD 10502413 EC50 = 0.8 nM T67162 CA1YR2 10502670 Ki = 4.94 nM T67162 CN9BT6 10512444 Ki = 2.5 nM T67162 C1NK6V 10515180 Ki = 779 nM T67162 CC4A7G 10515835 Ki = 4710 nM T67162 CN28AB 10515841 Ki = 74 nM T67162 C1GRL4 10518406 Ki = 1949.84 nM T67162 CL8R9O 10518820 Ki = 2980 nM T67162 CUQ03E 10520440 Ki = 900 nM T67162 CYL86S 10520941 Ki = 61 nM T67162 C2B9PT 10522146 Ki > 1600 nM T67162 C8ZMA1 10522334 Ki = 690 nM T67162 C12ZTU 10522613 Ki = 220 nM T67162 C38ACZ 10522614 Ki = 26 nM T67162 CYP98E 10522950 Ki = 12 nM T67162 C3EG1O 10524285 Ki = 1258.93 nM T67162 C7TZ3K 10524751 Ki = 5200 nM T67162 CQ5F3N 10525119 Ki = 398.11 nM T67162 CNO5P3 10527118 Ki = 403 nM T67162 CI67OK 10535587 Ki = 355 nM T67162 C3F0MU 10537661 Ki > 1000 nM T67162 CB7OK1 10541769 IC50 > 10000 nM T67162 C9ZYA3 10542345 Ki = 222 nM T67162 C4E6TV 10542381 Ki > 1600 nM T67162 C59NSH 10543696 Ki > 4130 nM T67162 C8ZG3C 10545941 Ki = 698 nM T67162 C48BRW 10546334 Ki = 1.66 nM T67162 CXI49Z 10546453 Ki = 150 nM T67162 C7UCS1 10546540 Ki = 95 nM T67162 CV57XZ 10546579 Ki = 1400 nM T67162 C40CJM 10546828 Ki = 240 nM T67162 CYF64N 10547607 Ki = 900 nM T67162 C23BRU 10548105 Ki > 5880 nM T67162 CKD0F6 10548329 Ki = 125.89 nM T67162 CQ2R5D 10548967 Ki = 3960 nM T67162 C4VZ2K 10549355 Ki > 1500 nM T67162 CU9CM3 10549689 EC50 = 2 nM T67162 C3P5VL 10550893 IC50 = 4.2 nM T67162 CQD6C8 10551026 Ki = 130 nM T67162 CBV9N4 10551197 Ki = 49 nM T67162 CH7E0W 10559624 Ki = 5.4 nM T67162 CKFH63 10560954 Ki = 254 nM T67162 CYCT15 10562462 Ki = 83.2 nM T67162 CVGI39 10564353 Ki = 30100 nM T67162 CSG18U 10566689 Ki > 1000 nM T67162 CJH5T9 10567430 Ki = 2500 nM T67162 C08LPE 10567839 Ki > 5800 nM T67162 C0HJS2 10568183 IC50 = 146 nM T67162 CB8VS9 10568394 Ki > 10000 nM T67162 CC56ON 10568805 Ki > 5800 nM T67162 CYL67U 10569690 Ki = 280 nM T67162 C60SMR 10570080 Ki = 83 nM T67162 CW38OC 10570563 Ki = 93 nM T67162 C6S0TG 10570898 Ki > 5800 nM T67162 CTR45A 10570997 Ki = 240 nM T67162 C5YH2I 10571274 Ki = 2030 nM T67162 C1YU3Q 10571927 Ki > 1500 nM T67162 CZ87BA 10572985 Ki = 980 nM T67162 CM3C1L 10573099 Ki > 850 nM T67162 CHE80N 10573876 Ki = 794.33 nM T67162 C02HSA 10574303 Ki = 8.8 nM T67162 CD3F9R 10575254 Ki = 125.89 nM T67162 CLT4X3 10585771 Ki > 1000 nM T67162 C0O6IU 10586728 Ki = 1530 nM T67162 C9SP3R 10587140 Ki = 650 nM T67162 COL98E 10588194 Ki = 251 nM T67162 CM97NV 10588666 Ki = 1600 nM T67162 CQ38ZC 10588763 Ki = 1010 nM T67162 CP1Y7K 10589218 Ki = 64 nM T67162 CT2R7G 10589834 IC50 > 10000 nM T67162 C8KND3 10589897 Ki > 1700 nM T67162 C12ZRK 10590285 Ki = 275.42 nM T67162 CEH05N 10590717 Ki = 536 nM T67162 C2M5PS 10591665 Ki > 1000 nM T67162 CRJ13B 10593191 Ki = 173.78 nM T67162 C7RXS4 10593347 Ki > 1000 nM T67162 C7EN0K 10593348 Ki = 2500 nM T67162 C8E4HR 10593869 Ki = 270 nM T67162 C97NMI 10594054 Ki = 220 nM T67162 CM7Z9X 10594113 Ki = 125 nM T67162 C17ZDI 10594242 Ki = 7.8 nM T67162 CTZ9V3 10594723 IC50 = 64 nM T67162 CD27FZ 10594764 Ki = 15 nM T67162 C1VLS4 10595646 Ki = 1584.89 nM T67162 CDO93P 10595908 Ki = 35 nM T67162 CA1B9Q 10596144 Ki = 2238.72 nM T67162 C57DKO 10596380 IC50 > 1000 nM T67162 CVZ10Y 10596978 Ki = 3.4 nM T67162 C9S0RY 10597050 Ki = 3400 nM T67162 CO23YX 10597140 Ki = 398.11 nM T67162 C6ECP0 10598935 Ki = 11 nM T67162 CU8DW9 10608413 Ki = 2450 nM T67162 C49WAM 10610641 Ki = 201 nM T67162 C6GB7W 10611439 Ki = 317 nM T67162 C7GDX0 10612157 Ki = 7.2 nM T67162 CH49UB 10613605 Ki = 107 nM T67162 C0D9FQ 10613676 Ki = 249 nM T67162 C74NSJ 10615016 Ki > 1600 nM T67162 C3FS5U 10615437 Ki = 66 nM T67162 CSI97L 10615684 Ki = 61 nM T67162 C9JI3A 10615787 Ki = 227 nM T67162 CB6HW4 10615990 IC50 = 68 nM T67162 C5XI7L 10616050 Ki = 1880 nM T67162 CPY43H 10617133 IC50 = 10 nM T67162 C56UGP 10617366 Ki = 90 nM T67162 CT5A6H 10617381 Ki = 48.98 nM T67162 CWQ76V 10617946 Ki = 960 nM T67162 C6QB8L 10618211 Ki = 120 nM T67162 C2LN0J 10618874 Ki = 520 nM T67162 CJ7R5F 10618875 Ki = 200 nM T67162 CPJ0H3 10618928 Ki = 4800 nM T67162 C3VQK1 10619612 Ki = 110 nM T67162 CJ40ZT 10619737 Ki = 290 nM T67162 CDZ16W 10620139 Ki > 5800 nM T67162 C1RXC5 10620194 Ki = 37 nM T67162 CX3A0P 10620719 Ki = 325 nM T67162 CD8KX9 10621491 Ki = 158 nM T67162 C6HAV3 10636896 Ki = 19.95 nM T67162 CKF8L2 10637198 Ki = 500 nM T67162 CKY6Z8 10637496 Ki = 411 nM T67162 C0V5NM 10638052 Ki = 118 nM T67162 C9PD7O 10639290 Ki > 50000 nM T67162 C8O4BC 10639430 Ki > 4130 nM T67162 CQ75TL 10640054 Ki > 1600 nM T67162 C8C2GN 10640055 Ki > 1600 nM T67162 C9D5MP 10640530 Ki = 1170 nM T67162 CK4O3W 10641637 Ki = 2600 nM T67162 C2B5NL 10641783 Ki > 5880 nM T67162 C89NYU 10641954 Ki > 5800 nM T67162 C0DCY3 10641955 Ki = 5500 nM T67162 CKP3A1 10642106 Ki > 5880 nM T67162 CPTF56 10642239 Ki = 451 nM T67162 CIFM84 10642428 Ki = 4.7 nM T67162 CT74PA 10643047 Ki = 46 nM T67162 CED15G 10643588 Ki = 170 nM T67162 CL8KB3 10643589 Ki = 73 nM T67162 CD21IV 10643697 IC50 > 1000 nM T67162 C4K0PA 10643780 Ki = 1400 nM T67162 C6TZS3 10644771 Ki = 2350 nM T67162 C0FTQ6 10656511 Ki = 82.3 nM T67162 C2W5BE 10660814 Ki = 61 nM T67162 CQM6J9 10662302 Ki = 3650 nM T67162 CFC38D 10663221 Ki = 3500 nM T67162 CTP8L0 10664621 Ki = 287 nM T67162 C43FER 10665101 Ki = 467.74 nM T67162 CU3XJ4 10665598 Ki = 540 nM T67162 CI2OT7 10665626 Ki = 659 nM T67162 CCU12E 10666005 IC50 = 17 nM T67162 C31ZOC 10666315 Ki = 52 nM T67162 CWE53T 10667201 Ki = 330 nM T67162 C7K9DP 10667579 Ki = 1300 nM T67162 C4IY3Z 10667966 Ki = 11000 nM T67162 CT45YR 10668173 IC50 = 7 nM T67162 CU14XK 10679285 Ki > 1000 nM T67162 CQ2F1P 10679847 Ki = 167 nM T67162 CU31PH 10682854 Ki = 5882 nM T67162 CO49AQ 10683127 Ki = 854 nM T67162 CN8AJ2 10683943 Ki = 311 nM T67162 C61IJT 10683945 Ki = 182 nM T67162 C01FQC 10684005 Ki > 10000 nM T67162 CZLJ52 10684706 Ki = 556 nM T67162 C0ZCG1 10684789 EC50 = 1 nM T67162 C6R7JD 10685891 Ki = 7 nM T67162 CZ08XG 10685957 Ki > 1000 nM T67162 C7T2FU 10687362 Ki > 5800 nM T67162 CJ6O7P 10687667 Ki > 1000 nM T67162 CY4Z1R 10687967 Ki = 310 nM T67162 CBW96O 10688035 Ki = 860 nM T67162 C60DRH 10688036 Ki = 900 nM T67162 C87BLK 10688561 IC50 = 128 nM T67162 CJFP08 10688858 IC50 = 56 nM T67162 CK0TC9 10688859 IC50 = 202 nM T67162 CMVD23 10689266 Ki > 5800 nM T67162 CC1E7W 10690200 Ki = 290 nM T67162 C75DXM 10690882 Ki = 10000 nM T67162 CEM56L 10691523 Ki = 700 nM T67162 CD1KF8 10691599 Ki = 130 nM T67162 CR2FI0 10691634 Ki = 398.11 nM T67162 C2LU1H 10692095 Ki = 386 nM T67162 CHZ8O2 10692886 Ki = 0.22 nM T67162 CS4JW5 10698929 Ki = 2260 nM T67162 C8OC6U 10704110 Ki = 0.67 nM T67162 C24FCX 10705905 Ki > 1000 nM T67162 CLZ9F5 10706553 Ki = 39.2 nM T67162 CBE87R 10706626 Ki = 261 nM T67162 C3DR0U 10707685 Ki = 26 nM T67162 CU25LW 10708280 Ki = 268 nM T67162 C49IUL 10708935 Ki > 1700 nM T67162 C2ZJH4 10709505 Ki > 1000 nM T67162 C52SWI 10711404 Ki > 1600 nM T67162 CV9S1L 10712078 Ki = 39 nM T67162 C49QRP 10712278 Ki > 1000 nM T67162 CN6E5P 10713210 Ki > 5000 nM T67162 CSXO03 10713599 IC50 = 32 nM T67162 CE5QA3 10713620 Ki = 2.2 nM T67162 C7PDA6 10713670 Ki = 500 nM T67162 CG8KF5 10713960 Ki = 25 nM T67162 C4O6KG 10714184 Ki = 410 nM T67162 CIQ45P 10715225 Ki > 850 nM T67162 CA8MK0 10715375 Ki = 3162.28 nM T67162 CCW26V 10715828 EC50 = 0.3 nM T67162 C0USP7 10718592 Ki > 1000 nM T67162 CHN8Q9 10725712 Ki = 585 nM T67162 CHN3T8 10729313 Ki = 26 nM T67162 CQU83R 10730269 Ki = 23.8 nM T67162 C5DIW2 10732337 Ki = 1750 nM T67162 C71VBX 10732925 Ki = 295.12 nM T67162 CWY6V1 10733406 Ki = 21.88 nM T67162 CO9BL7 10734727 Ki = 245 nM T67162 CHN4A3 10735344 Ki > 1900 nM T67162 CQ2DU0 10735405 Ki = 82 nM T67162 CO1DT0 10735463 Ki = 1440 nM T67162 C3L7EO 10736014 Ki = 1330 nM T67162 C8VGB5 10736673 Ki = 5.7 nM T67162 CJM1R5 10737150 Ki = 2740 nM T67162 CNWC38 10737474 Ki = 66.07 nM T67162 CY5HG9 10738530 Ki = 560 nM T67162 CSA67W 10738750 Ki = 8.5 nM T67162 C65DWL 10739194 IC50 = 228 nM T67162 CI06WV 10740593 Ki = 3.2 nM T67162 C6PED3 10754042 Ki = 215 nM T67162 C4I9VE 10756932 Ki = 2400 nM T67162 CP83GM 10757141 Ki = 238 nM T67162 C9Z8TB 10757990 Ki > 3500 nM T67162 C8XD2C 10758004 Ki = 1318.26 nM T67162 C19UPY 10759511 Ki > 5800 nM T67162 C21TFA 10759963 Ki = 5.7 nM T67162 CH5AY1 10760638 Ki = 602.56 nM T67162 CHN8T2 10760813 Ki = 120 nM T67162 C9FE7Z 10761040 IC50 = 2 nM T67162 CDNE69 10761258 Ki = 363.08 nM T67162 CAV6N0 10761912 Ki = 282 nM T67162 CC2L1A 10762432 Ki = 60 nM T67162 C3TD1I 10762475 Ki = 31.62 nM T67162 CAO80C 10762881 Ki > 1300 nM T67162 C80STM 10763496 Ki = 262 nM T67162 C5WH2F 10763756 EC50 = 0.8 nM T67162 CAWG43 10765237 Ki = 6 nM T67162 CZ3M9J 10777894 Ki > 10000 nM T67162 CQ2R0A 10780076 IC50 = 263 nM T67162 C3LB9N 10780510 Ki = 143 nM T67162 CX4NK7 10780717 EC50 = 9.8 nM T67162 C1RG2E 10780842 Ki = 7980 nM T67162 CRUD74 10780928 Ki = 47 nM T67162 CU9T8V 10780942 Ki = 112 nM T67162 C2MPX6 10782049 Ki = 352 nM T67162 CIDM49 10782111 IC50 = 171 nM T67162 C6D3BX 10783358 Ki > 1000 nM T67162 C4G8HB 10783874 Ki = 11 nM T67162 C1K4OD 10785202 Ki = 180 nM T67162 C6JT9I 10786190 Ki = 195 nM T67162 C6J2FC 10786367 Ki = 570 nM T67162 CF9S6Q 10786474 Ki > 850 nM T67162 CCBO47 10786591 Ki > 5800 nM T67162 C96NIC 10786891 Ki = 6 nM T67162 CXO6J4 10801405 Ki = 3351 nM T67162 CL1CV6 10801925 Ki = 228 nM T67162 CJK8L2 10803661 Ki = 2760 nM T67162 C46LYA 10803754 IC50 = 766 nM T67162 CP74YO 10803828 Ki = 2.5 nM T67162 CB74KW 10803829 Ki = 73.9 nM T67162 CEM9Y6 10804534 Ki > 1600 nM T67162 CFH1Q4 10805130 Ki > 1600 nM T67162 CB45KG 10805355 Ki = 1400 nM T67162 CZ7J1S 10805599 Ki = 70.8 nM T67162 CT5XK8 10805917 Ki > 10000 nM T67162 C5M9AW 10806501 Ki = 1300 nM T67162 CNWV56 10807035 Ki = 1170 nM T67162 CWA5J0 10807321 Ki > 1000 nM T67162 CS7YU8 10807795 Ki = 610 nM T67162 CRZU91 10808230 IC50 = 5 nM T67162 CGVU78 10808677 Ki > 10000 nM T67162 C24QAM 10809899 Ki = 38 nM T67162 CS0BT5 10810976 Ki = 3170 nM T67162 C9JR8A 10811378 EC50 = 5 nM T67162 C1VTJ3 10811814 Ki > 850 nM T67162 CZ1F3B 10824155 Ki = 12000 nM T67162 CU32QP 10825256 Ki = 183 nM T67162 CUI27T 10825325 Ki = 19.4 nM T67162 C1SK9V 10826290 Ki > 590 nM T67162 C75SRI 10826543 Ki = 2050 nM T67162 CJ9BY0 10827222 EC50 = 1.7 nM T67162 CN0S5A 10827592 Ki = 1000 nM T67162 CE7M9P 10829708 IC50 = 5 nM T67162 CCN52S 10830557 Ki = 1800 nM T67162 CK92FA 10831286 Ki > 10000 nM T67162 C1QMR4 10831735 Ki = 7600 nM T67162 CJ1DI4 10831786 Ki = 3400 nM T67162 CL4T8O 10832341 Ki = 5000 nM T67162 C4R7DC 10832895 IC50 = 810 nM T67162 CM83SE 10833953 Ki = 36000 nM T67162 C8MHZ9 10835110 Ki = 1000 nM T67162 CDB9X1 10849018 Ki = 177 nM T67162 C3GR4Q 10850084 Ki > 1000 nM T67162 C14VQN 10851217 IC50 = 37 nM T67162 CQRA27 10851283 Ki > 1000 nM T67162 CDOH18 10851309 Ki > 1600 nM T67162 CF1S7E 10852461 Ki = 190 nM T67162 C0VQ3C 10853014 Ki > 1600 nM T67162 CNPB35 10854042 EC50 = 54.95 nM T67162 CPU26G 10854370 Ki = 52.5 nM T67162 CI6PW4 10854386 Ki = 110 nM T67162 C53OXZ 10861560 Ki > 1000 nM T67162 CV6ZN3 10861900 Ki > 1000 nM T67162 C9A8KN 10862425 Ki = 84 nM T67162 CHS8N5 10862670 Ki = 66.8 nM T67162 CL9Q3F 10863645 Ki = 178 nM T67162 CZYF05 10871118 Ki = 16000 nM T67162 C20CTE 10873003 Ki = 2 nM T67162 C1UQ4H 10873318 Ki = 253 nM T67162 CKOF21 10873956 Ki = 63 nM T67162 CJ17GX 10874342 Ki = 18 nM T67162 CQ3TR7 10879566 Ki = 2037 nM T67162 CMV36C 10884046 Ki = 65 nM T67162 CLEM91 10885047 Ki = 94.6 nM T67162 CD3U9P 10885524 Ki = 10 nM T67162 CRI50E 10885636 IC50 = 2240 nM T67162 CNP08C 10891703 Ki > 10000 nM T67162 CL4S8G 10893228 Ki = 19117 nM T67162 CV4ZO0 10894526 Ki = 14.5 nM T67162 CU80EA 10895106 Ki = 35 nM T67162 CMJD46 10895845 Ki = 21 nM T67162 CW8UH1 10905430 Ki = 13 nM T67162 C8CZB9 10905940 Ki = 1130 nM T67162 C3X6QE 10906470 Ki = 128 nM T67162 CCHK19 10906679 Ki = 23 nM T67162 CX65PW 10907460 IC50 = 2890 nM T67162 CSM1Q2 10919602 Ki = 7.2 nM T67162 CDR7G5 10925892 Ki = 1000 nM T67162 CNT3E2 10926404 Ki > 1000 nM T67162 C9OI8S 10927262 Ki > 1500 nM T67162 C67FYJ 10927750 Ki = 825 nM T67162 CN7C6W 10927912 Ki = 20.9 nM T67162 CH2OW6 10928654 Ki = 50.2 nM T67162 C7AKH6 10939008 Ki = 23 nM T67162 CGZA42 10939167 EC50 = 12 nM T67162 C0UGV5 10939222 Ki = 39.81 nM T67162 C69ULE 10939408 Ki = 1149 nM T67162 CPBA97 10939644 Ki = 23.7 nM T67162 C25TSY 10940279 Ki = 63 nM T67162 CC07JE 10942784 Ki = 3.3 nM T67162 CNB39C 10947658 Ki = 60 nM T67162 CN7XS4 10948527 IC50 = 557 nM T67162 CO7P5V 10948748 Ki > 1000 nM T67162 C2SMP6 10949917 Ki = 14 nM T67162 C0WX2Y 10950176 Ki = 1410 nM T67162 CVN2Y8 10950916 Ki = 235 nM T67162 C1JD5K 10951105 Ki = 68 nM T67162 CJ5HP9 10951185 Ki = 32 nM T67162 C3JCI2 10960333 Ki = 37000 nM T67162 C2IGR9 10960767 Ki = 19 nM T67162 CBPS24 10961112 Ki = 10.3 nM T67162 CH14OY 10961938 Ki = 830 nM T67162 CUNX16 10971014 Ki = 11.1 nM T67162 C4PK7X 10971209 Ki = 1500 nM T67162 C9DLO4 10971923 Ki = 26.5 nM T67162 C9HPJ3 10972865 Ki = 2570 nM T67162 CE5PG3 10974122 Ki = 103 nM T67162 C6NF4A 10978080 Ki = 794.33 nM T67162 CFU1S9 10980338 Ki = 13000 nM T67162 C2HP7F 10981761 IC50 = 123 nM T67162 CJL0F7 10983103 Ki = 145 nM T67162 CB86ST 10983150 Ki = 11 nM T67162 CM9JY3 10988746 Ki = 3107 nM T67162 C0BUR1 10991521 Ki = 750 nM T67162 C9AIQ2 10993488 Ki = 330 nM T67162 CWQ40B 10994141 Ki = 430 nM T67162 CNU2H3 10994539 Ki = 114 nM T67162 CS72LE 10994916 Ki = 161 nM T67162 C0FV9Z 11003833 Ki = 680 nM T67162 CY3KA2 11005177 Ki = 56 nM T67162 CJC9K4 11005810 IC50 = 551 nM T67162 CO36VS 11005852 Ki = 5 nM T67162 CE6HJ8 11013863 Ki = 710 nM T67162 C6GT4A 11014340 Ki = 57.54 nM T67162 CN32LJ 11015257 Ki = 44 nM T67162 C3FWN7 11016080 Ki = 45 nM T67162 C6BZR9 11016169 Ki = 63 nM T67162 CXZ29Y 11016342 Ki > 1000 nM T67162 CT56RB 11026289 Ki = 777 nM T67162 CGHN43 11027407 Ki = 15.2 nM T67162 CQ6M1S 11028157 Ki = 3800 nM T67162 CJ15OI 11036114 Ki > 1000 nM T67162 CG9JC8 11036563 Ki = 680 nM T67162 C01NDT 11036640 Ki = 150 nM T67162 CU6HR7 11036641 Ki = 3.9 nM T67162 C7C2RI 11044146 Ki = 439 nM T67162 C7KDU9 11048013 Ki = 56 nM T67162 CQ97YN 11048095 Ki = 11.5 nM T67162 C0N9VE 11048899 Ki = 200 nM T67162 C9FPV0 11048937 Ki = 200 nM T67162 CL5DF2 11057472 Ki = 650 nM T67162 C0SUF4 11057969 Ki = 85 nM T67162 C9ZGU6 11058213 Ki = 1100 nM T67162 CTL9P3 11058442 Ki = 9.5 nM T67162 CT9CZ1 11058829 Ki = 892 nM T67162 CE3J0B 11068912 Ki = 480 nM T67162 CP21DQ 11069795 Ki = 10 nM T67162 CG41BK 11071079 IC50 = 2620 nM T67162 CVCE26 11076818 Ki = 1080 nM T67162 CG63OS 11077918 Ki = 31000 nM T67162 CNF43K 11078813 Ki = 39000 nM T67162 CGEY62 11079151 Ki = 1100 nM T67162 CE85YF 11079832 Ki = 635 nM T67162 C9LCB6 11090403 Ki > 1000 nM T67162 CQ6W8Y 11091160 Ki = 12 nM T67162 CFI32S 11095339 Ki > 10000 nM T67162 CL7AX5 11099801 Ki > 1500 nM T67162 CP4WL3 11100243 Ki = 1800 nM T67162 C76FKX 11100514 Ki = 490 nM T67162 CN43SG 11102013 EC50 = 10 nM T67162 C6TAH5 11102080 Ki = 35 nM T67162 CBM1I9 11102188 Ki = 8 nM T67162 C94EVP 11102206 Ki = 14 nM T67162 CW83IO 11102301 Ki = 32 nM T67162 CO5Y6W 11113582 Ki = 117 nM T67162 C4HK6I 11120635 Ki > 1500 nM T67162 CVE8T3 11121216 Ki = 330 nM T67162 CUN87A 11122812 Ki = 15 nM T67162 CVM23D 11123162 Ki = 107 nM T67162 C8TW2P 11131951 Ki = 7460 nM T67162 CHX96W 11133309 Ki = 650 nM T67162 CTXS48 11133385 Ki = 606 nM T67162 CWG8O0 11133533 Ki = 770 nM T67162 CXP12A 11133602 Ki = 7.1 nM T67162 CUD5A0 11134444 Ki = 113 nM T67162 C0C3FI 11134596 Ki = 126 nM T67162 C2API9 11141325 Ki = 530 nM T67162 CWT4S5 11144835 Ki = 1560 nM T67162 CQC54U 11145409 Ki = 630 nM T67162 CK7H9L 11146824 Ki = 729 nM T67162 CHD24Z 11151081 EC50 > 10000 nM T67162 C9MWB5 11151919 EC50 > 10000 nM T67162 CEX52K 11151920 Ki = 68 nM T67162 CWC6E8 11152302 Ki > 1000 nM T67162 C3Q9UG 11154178 Ki = 159 nM T67162 CNE31P 11163137 EC50 > 10000 nM T67162 CW7Y9O 11163741 Ki = 794.33 nM T67162 C4K6QP 11164276 Ki = 132 nM T67162 C56VFO 11166027 Ki = 18.2 nM T67162 CAY3B5 11175544 Ki = 97 nM T67162 CQ7ZA0 11175610 EC50 > 10000 nM T67162 C75WKP 11176199 IC50 = 44 nM T67162 C39PED 11177610 Ki = 6.6 nM T67162 C6CL1Y 11178830 Ki = 1258.93 nM T67162 C0W4SM 11186523 Ki = 12 nM T67162 CN06GJ 11186895 Ki = 42.4 nM T67162 C3CIH1 11187957 EC50 > 10000 nM T67162 C9CTH8 11188446 Ki > 1000 nM T67162 CSQH27 11191128 Ki = 987 nM T67162 CG7D2K 11198974 EC50 > 10000 nM T67162 C8PF9M 11199162 Ki = 63.8 nM T67162 C4CW6X 11200205 Ki = 64.5 nM T67162 C9N5QU 11200511 Ki > 2000 nM T67162 CP8ZQ6 11203357 Ki = 28.1 nM T67162 CPX23W 11209208 IC50 > 10000 nM T67162 C4J8YG 11211017 Ki = 2200 nM T67162 CI0M3S 11211058 Ki = 995 nM T67162 CXO67U 11213037 Ki = 128.82 nM T67162 C41FWO 11213062 Ki = 1 nM T67162 CQ1E8L 11213136 Ki = 79.43 nM T67162 C6V2QH 11221906 Ki = 137 nM T67162 CEFK20 11222637 EC50 > 10000 nM T67162 C6RXG7 11222979 Ki > 1000 nM T67162 C6D1MZ 11223004 Ki > 5000 nM T67162 C8RJ3D 11223303 Ki = 6000 nM T67162 CN7CG0 11224283 Ki = 30.4 nM T67162 C1VM2S 11225043 Ki = 100 nM T67162 CA39QR 11227406 IC50 = 1000 nM T67162 C6LB4S 11230330 Ki = 130 nM T67162 CF42AW 11233507 Ki = 1.51 nM T67162 CKX06B 11235174 Ki = 3000 nM T67162 CCKI68 11247894 Ki = 21.9 nM T67162 C7RW8Y 11248332 Ki = 265 nM T67162 C90WSG 11248705 Ki = 1258.93 nM T67162 CHQ8X4 11249540 Ki = 10.6 nM T67162 CL04EZ 11256262 Ki = 128 nM T67162 CH92LP 11256583 EC50 > 10000 nM T67162 C7BG9T 11258233 Ki = 19.6 nM T67162 C7XI0R 11260032 Ki = 501.19 nM T67162 C8JW3Z 11260311 Ki = 291 nM T67162 CU8HM2 11268785 Ki = 45.5 nM T67162 CM72YX 11269330 Ki = 756 nM T67162 CD47FC 11269392 EC50 > 10000 nM T67162 CC0YP2 11271099 Ki = 19.95 nM T67162 CL0DP6 11272440 Ki = 630.96 nM T67162 C4S2VF 11277147 Ki > 1000 nM T67162 C27GXZ 11277680 IC50 > 10000 nM T67162 CKN4L3 11280225 EC50 > 10000 nM T67162 CUJ2R7 11280344 Ki = 383 nM T67162 CZG20K 11281627 Ki = 6.1 nM T67162 C48WZU 11282073 Ki = 10.2 nM T67162 CY6MX5 11282296 Ki = 68 nM T67162 CP0R9A 11283795 Ki > 1000 nM T67162 C8LAP9 11292299 EC50 > 10000 nM T67162 CC2Y4X 11299620 Ki = 6 nM T67162 C57GTA 11299968 IC50 > 10000 nM T67162 C2ABW4 11301354 EC50 > 10000 nM T67162 C9BLC7 11304596 Ki = 794.33 nM T67162 CJS9C0 11304851 IC50 > 3200 nM T67162 CIMB79 11305766 Ki = 398.11 nM T67162 C1PDJ5 11306892 Ki = 566 nM T67162 C4DSN3 11307083 Ki = 35.4 nM T67162 CI79LV 11307899 Ki = 3.162 nM T67162 CUXZ91 11311148 IC50 > 10000 nM T67162 C2GZD3 11311204 IC50 > 10000 nM T67162 CSA7U3 11313751 Ki = 7.53 nM T67162 CI56TH 11314352 EC50 > 10000 nM T67162 C5K8SP 11314647 Ki = 44.8 nM T67162 CU82GC 11315254 Ki = 7.06 nM T67162 C85FPO 11315462 Ki > 10000 nM T67162 CU2GF6 11316078 Ki = 29 nM T67162 CXC2R6 11316847 EC50 = 13.8 nM T67162 C6FD1Z 11317018 Ki = 65.5 nM T67162 C9RW3C 11324794 Ki = 172 nM T67162 CIZH05 11325334 Ki = 168 nM T67162 CP5AF8 11325645 EC50 > 10000 nM T67162 CF38AZ 11325818 EC50 > 10000 nM T67162 CJ2TH8 11326248 Ki > 1000 nM T67162 CSR03X 11326600 Ki = 13.2 nM T67162 CH35RX 11327651 Ki = 10.1 nM T67162 C3FSK5 11329254 Ki = 681 nM T67162 CIK35D 11336814 Ki = 46.6 nM T67162 CTIX74 11338096 Ki = 2850 nM T67162 CRMK35 11338674 Ki = 31.2 nM T67162 CGB7I6 11341394 Ki > 1000 nM T67162 C0NRE8 11346967 Ki = 5317 nM T67162 CPA4W3 11349297 Ki > 1000 nM T67162 C4XC2F 11349635 Ki = 105 nM T67162 CJT5E1 11350623 Ki > 1000 nM T67162 CCY23Q 11351639 Ki = 149 nM T67162 CX7S0U 11352111 Ki = 43.7 nM T67162 CA1NC6 11356479 Ki = 160 nM T67162 CXWH42 11358377 Ki > 10000 nM T67162 CCVK79 11370781 Ki = 1820 nM T67162 CBPJ98 11371795 EC50 > 10000 nM T67162 CY24NV 11374299 Ki = 2000 nM T67162 CUC3D2 11382826 Ki = 1.738 nM T67162 COD89G 11383046 Ki > 1000 nM T67162 CBV52J 11384146 Ki > 2000 nM T67162 C1OM3C 11384207 Ki = 467.74 nM T67162 CO1I8H 11384634 Ki = 22 nM T67162 C4SZ7W 11384664 Ki = 238 nM T67162 CT1SY6 11385992 Ki = 51 nM T67162 CPQU06 11393136 Ki > 1000 nM T67162 CFN86P 11394557 Ki = 1.3 nM T67162 CGJ2Z7 11394708 EC50 > 10000 nM T67162 CQ5BN6 11396088 Ki = 8.8 nM T67162 C9AOM3 11397017 Ki = 199.53 nM T67162 CF4OX6 11397149 Ki = 79.43 nM T67162 C82ERW 11397777 Ki = 251.19 nM T67162 C1V4EQ 11404156 Ki > 10000 nM T67162 CDV4A0 11405107 Ki = 550 nM T67162 CT32OJ 11406143 Ki = 4188 nM T67162 C3OL9U 11406615 Ki = 2.75 nM T67162 C2ZCG3 11407062 Ki = 16.9 nM T67162 CGN10L 11408148 Ki = 76.5 nM T67162 C1XD0I 11408287 Ki = 7.4 nM T67162 CJUI62 11416883 EC50 > 10000 nM T67162 CV1AT8 11417923 Ki > 1000 nM T67162 CFX98O 11418182 Ki = 310 nM T67162 C91RNU 11419120 Ki = 39.1 nM T67162 CLH0N1 11429008 Ki = 33 nM T67162 C85LYP 11430418 IC50 > 100 nM T67162 C6K5MH 11431530 Ki = 1000 nM T67162 CO6F2D 11431895 Ki = 217 nM T67162 CNF28A 11432177 Ki = 26.4 nM T67162 CBN91Q 11439190 Ki = 1328 nM T67162 C6S1FL 11442000 Ki = 17.5 nM T67162 CU3A2F 11442772 Ki = 8 nM T67162 CTM1W8 11443078 Ki = 18.2 nM T67162 CY1M6Q 11450607 EC50 > 10000 nM T67162 C86CJB 11451022 Ki = 219 nM T67162 CF6AM3 11451082 Ki = 0.67 nM T67162 CA3JG1 11451703 Ki = 171 nM T67162 C6SVK9 11452692 Ki = 54.5 nM T67162 C0TKD2 11452896 Ki = 5.8 nM T67162 CB3P6S 11452916 Ki = 3300 nM T67162 C05VEA 11453253 Ki = 281.84 nM T67162 CTA58W 11469395 Ki = 334 nM T67162 C8L6ZI 11472028 Ki = 6280 nM T67162 C3MJK9 11474718 Ki > 1000 nM T67162 CLZ91D 11474734 EC50 > 10000 nM T67162 C3GMQ1 11477018 Ki = 630.96 nM T67162 C4V1MG 11477201 Ki = 45.7 nM T67162 C2HU6O 11480902 Ki = 4890 nM T67162 CK39HZ 11486421 Ki = 3900 nM T67162 C5HVS4 11486446 Ki = 0.05248 nM T67162 CYZ79A 11486571 Ki = 26.1 nM T67162 CQL8F0 11487016 Ki = 5.94 nM T67162 CFE98H 11487464 Ki = 15 nM T67162 CTU1Z7 11488247 Ki = 331 nM T67162 C8BY4A 11489501 Ki > 794.33 nM T67162 C4TWQ0 11493559 IC50 > 10000 nM T67162 CKV25P 11493746 Ki = 37.5 nM T67162 C57LEG 11493794 IC50 = 5300 nM T67162 C8FN2P 11494093 Ki > 1000 nM T67162 CVLF59 11495417 Ki = 35.7 nM T67162 C9TU8S 11495769 Ki = 1.4 nM T67162 COI68V 11496213 Ki = 0.59 nM T67162 CPX26I 11496746 Ki > 794.33 nM T67162 CNC9V7 11496793 Ki > 1000 nM T67162 C5Z7GQ 11497411 Ki > 501.19 nM T67162 C9YU1O 11497679 Ki < 1584.89 nM T67162 CQT5U8 11497680 Ki > 794.33 nM T67162 C9JD4N 11497924 Ki > 1000 nM T67162 CR1HO4 11500181 Ki > 10000 nM T67162 CAU1R7 11500677 Ki = 21.1 nM T67162 CASD80 11501253 Ki > 1000 nM T67162 C16AXW 11501537 Ki > 1000 nM T67162 C3ROH5 11504077 Ki = 15.85 nM T67162 CN84HD 11504199 Ki = 130 nM T67162 CN63TR 11504230 Ki = 5.6 nM T67162 CTMH12 11505007 Ki = 114 nM T67162 CXE65Q 11505572 Ki > 750 nM T67162 C16TWK 11508052 IC50 > 10000 nM T67162 CRDF59 11509984 Ki = 179 nM T67162 CF45XR 11511026 Ki = 0.6 nM T67162 COT4H9 11511117 Ki > 794.33 nM T67162 C9BT2W 11512263 Ki = 1.5 nM T67162 C7FH8P 11512962 Ki = 1246 nM T67162 C59SCV 11516033 Ki = 2700 nM T67162 CRPD50 11517423 Ki = 5.3 nM T67162 CAMP52 11517928 Ki = 710 nM T67162 CQ0IF2 11518499 Ki > 1000 nM T67162 CJ0B8E 11518546 Ki > 750 nM T67162 CZ3D5Y 11518933 Ki > 2511.89 nM T67162 C0WU7G 11518972 Ki > 125.89 nM T67162 CM4B3J 11519133 Ki < 501.19 nM T67162 C08JSL 11519134 Ki > 501.19 nM T67162 CS20NG 11519153 Ki = 133 nM T67162 C04RCG 11519858 Ki > 2511.89 nM T67162 CXWO08 11522273 IC50 > 10000 nM T67162 CQ5IN9 11522339 Ki = 7.9 nM T67162 CC6U7R 11522476 Ki > 5000 nM T67162 C0WI4V 11523930 Ki = 90 nM T67162 C13YVG 11524412 Ki = 15.5 nM T67162 CO95XH 11525938 Ki = 501.19 nM T67162 CTNX29 11526451 Ki > 398.11 nM T67162 CR9NA7 11526531 Ki > 630.96 nM T67162 CNL15V 11527195 Ki > 1584.89 nM T67162 C38QFE 11530118 IC50 > 10000 nM T67162 CJF92G 11533429 Ki > 794.33 nM T67162 C2EQ1U 11533448 Ki < 398.11 nM T67162 C4LOQ9 11533473 Ki < 398.11 nM T67162 CZW9U3 11534726 Ki > 1584.89 nM T67162 C75YUO 11536580 Ki > 10000 nM T67162 C2JT3I 11536995 Ki = 39.9 nM T67162 C7DBO0 11537385 Ki > 1000 nM T67162 C07QHM 11539056 Ki = 1 nM T67162 CSN91H 11539722 Ki > 501.19 nM T67162 C0X6CJ 11540474 Ki < 1584.89 nM T67162 CO0R2G 11540842 Ki = 10 nM T67162 CN3W7S 11543350 Ki > 10000 nM T67162 C8X0EM 11543992 Ki > 10000 nM T67162 CMJ1B4 11545687 Ki = 14.6 nM T67162 C5ZY6N 11545813 Ki = 178.4 nM T67162 C7QKD5 11547151 Ki = 35 nM T67162 CD14OF 11547466 Ki > 630.96 nM T67162 CO5GF0 11547643 Ki = 519 nM T67162 C61LDE 11548217 Ki > 630.96 nM T67162 CKZ9B0 11548239 Ki < 316.23 nM T67162 CPA7K8 11548755 Ki = 630.96 nM T67162 C0AN1Y 11551474 Ki ~ 500 nM T67162 C9VC7O 11551780 IC50 > 10000 nM T67162 CA5G2Q 11552027 Ki = 62 nM T67162 C0ZD8A 11552981 Ki = 10.6 nM T67162 CBK1V7 11553516 Ki = 7.4 nM T67162 CW17TM 11554167 Ki = 1.2 nM T67162 C0ZBJ6 11554490 Ki = 1 nM T67162 C9XJP4 11554548 Ki = 501.19 nM T67162 CHDO61 11554831 Ki = 56.6 nM T67162 CBD05S 11554891 Ki > 750 nM T67162 C0VMG7 11555265 Ki > 630.96 nM T67162 C3Y4GR 11555971 Ki > 630.96 nM T67162 C7S2WZ 11558055 Ki = 17.38 nM T67162 CM8G3B 11558247 Ki = 26.1 nM T67162 C4HDA6 11558324 Ki > 10000 nM T67162 C1V5CH 11559090 Ki > 10000 nM T67162 CY5I0U 11559581 Ki = 8200 nM T67162 C9UH2M 11559589 Ki = 980 nM T67162 C4LEF8 11560215 Ki = 10.7 nM T67162 CH67TN 11560697 Ki = 2.3 nM T67162 C4N0JC 11561601 Ki = 630.96 nM T67162 CX1VD8 11562113 Ki > 501.19 nM T67162 C0JU9T 11562199 Ki < 199.53 nM T67162 C4N8JS 11562200 Ki > 794.33 nM T67162 C8GK0U 11566745 Ki = 65.7 nM T67162 CVP1Q9 11567578 Ki = 286 nM T67162 CEV2P7 11567620 Ki = 1.5 nM T67162 CD3Z7J 11567928 Ki > 1000 nM T67162 CG7VZ5 11568232 Ki = 27.2 nM T67162 CUH8Y7 11568543 Ki > 750 nM T67162 C52PDV 11568714 Ki > 1000 nM T67162 CR7M5S 11568725 Ki = 0.55 nM T67162 CNH1K4 11568826 Ki = 1.2 nM T67162 C0V5IK 11569099 Ki > 750 nM T67162 CCO29B 11569488 Ki > 750 nM T67162 C5J2UP 11569619 Ki = 14 nM T67162 CU6EY8 11569996 Ki = 398.11 nM T67162 CRK97Z 11570471 Ki = 3 nM T67162 C32JGN 11570589 Ki = 0.91 nM T67162 CP8MF4 11573628 Ki = 2 nM T67162 C1TBC8 11573806 Ki = 0.62 nM T67162 CTG5X1 11574902 Ki = 130 nM T67162 CA3D4I 11574985 Ki = 8.7 nM T67162 C8NMI4 11575479 Ki > 10000 nM T67162 C1Q8LC 11575799 Ki = 3500 nM T67162 C84MJZ 11576059 Ki = 1995.26 nM T67162 CASH81 11576387 Ki > 316.23 nM T67162 CE60FY 11576528 Ki = 2.5 nM T67162 C8YLD3 11577158 Ki < 1000 nM T67162 CZEB03 11577696 Ki = 141 nM T67162 CR8E2F 11578028 Ki > 1000 nM T67162 C6JC2T 11580039 IC50 > 10000 nM T67162 C8CU1X 11581237 Ki = 79 nM T67162 C4BGF8 11581443 Ki = 90 nM T67162 CM4H5G 11581611 Ki = 17.9 nM T67162 C9LH5J 11582322 Ki = 2.1 nM T67162 CQ09NJ 11583188 Ki = 72 nM T67162 C0HFP7 11584185 Ki > 1258.93 nM T67162 CS1OR8 11584530 Ki = 0.76 nM T67162 C6D1MA 11584660 Ki = 316.23 nM T67162 CU4J2W 11584694 Ki = 501.19 nM T67162 CI2FK6 11584858 Ki = 0.58 nM T67162 CN5DQ9 11585034 Ki > 630.96 nM T67162 C73UHS 11585248 Ki = 398.11 nM T67162 C3N4JH 11588926 Ki = 21 nM T67162 C1M2CP 11589069 Ki = 960 nM T67162 C3V6LN 11590801 Ki = 1.6 nM T67162 CC75MD 11590828 Ki > 794.33 nM T67162 CYX50J 11591601 Ki > 794.33 nM T67162 CIUL60 11591633 Ki > 630.96 nM T67162 CU45DK 11595209 Ki > 10000 nM T67162 C5Q8XM 11595240 Ki = 0.13 nM T67162 CW7C4E 11596369 Ki = 19 nM T67162 C1TOP5 11598123 Ki > 794.33 nM T67162 CFC25K 11601627 Ki > 10000 nM T67162 C6G7WS 11603119 Ki > 1000 nM T67162 CGD62Y 11603486 Ki = 5596 nM T67162 C02PTV 11603842 Ki = 9.1 nM T67162 CU2V5R 11603959 Ki = 86.2 nM T67162 C9L3NI 11605088 Ki > 750 nM T67162 C9DI6R 11606176 Ki > 501.19 nM T67162 CO1A5Z 11606378 Ki < 794.33 nM T67162 CL04ZJ 11606435 Ki > 630.96 nM T67162 CJC5N8 11606456 Ki > 1000 nM T67162 CZPE61 11608015 Ki = 5825 nM T67162 C7KA3R 11610248 Ki = 45 nM T67162 C2AFI7 11611862 Ki = 369 nM T67162 C9VOB8 11613105 Ki = 2.7 nM T67162 CYR7B5 11613115 Ki = 5.1 nM T67162 CT16JP 11613587 Ki > 630.96 nM T67162 CN91SZ 11613873 Ki > 630.96 nM T67162 C9BZG0 11615489 Ki = 4.6 nM T67162 C62SOL 11615782 Ki > 20000 nM T67162 C9D7OU 11616435 Ki > 10000 nM T67162 C7XB8E 11618408 Ki = 31 nM T67162 CKB59U 11620847 Ki > 1584.89 nM T67162 CXY07A 11621352 Ki < 316.23 nM T67162 CN1P4I 11623343 Ki = 19 nM T67162 CIZ53S 11623652 Ki ~ 100 nM T67162 CB7M8E 11625642 Ki > 1000 nM T67162 CC2G9I 11626748 Ki = 7800 nM T67162 C9FSA8 11627847 Ki > 1258.93 nM T67162 C51IBH 11627879 Ki > 2511.89 nM T67162 CE8W1Z 11628452 Ki > 501.19 nM T67162 CFJN71 11628631 Ki > 398.11 nM T67162 C8R6MK 11630058 Ki > 100000 nM T67162 CS4CR7 11631304 Ki > 5000 nM T67162 C8ZU2X 11631892 Ki = 2700 nM T67162 CGWO53 11632952 Ki = 24 nM T67162 C7CZE3 11633170 Ki = 100 nM T67162 CMX4K8 11633643 Ki > 10000 nM T67162 C2YHQ0 11633739 Ki = 1.7 nM T67162 CMZR85 11633816 Ki = 418 nM T67162 C5W0JR 11633992 Ki = 13 nM T67162 CG1C3D 11637457 Ki = 92 nM T67162 C2OU7Y 11638332 Ki > 10000 nM T67162 C19UMY 11638640 Ki > 1000 nM T67162 CI17EA 11638780 Ki = 9900 nM T67162 C35WZF 11639064 Ki = 3.8 nM T67162 CH89AK 11639248 Ki > 1000 nM T67162 C0XC2N 11641596 Ki > 2511.89 nM T67162 C25KGE 11641641 Ki < 501.19 nM T67162 C8DXS0 11642163 Ki < 398.11 nM T67162 CLZQ65 11644613 Ki > 10000 nM T67162 CEN25S 11646648 Ki = 5.5 nM T67162 CMIC92 11647002 EC50 > 10000 nM T67162 CT72XD 11647101 Ki = 1 nM T67162 C9YA0E 11647443 Ki = 1 nM T67162 CYQB50 11648990 Ki > 630.96 nM T67162 C9XD0H 11649431 Ki = 6.4 nM T67162 CEZO71 11652518 Ki = 49000 nM T67162 CHIW07 11652965 Ki > 10000 nM T67162 C1HDM5 11653679 Ki = 43.3 nM T67162 CJV2I4 11655403 Ki = 1.1 nM T67162 C5T4UV 11655570 Ki = 88 nM T67162 C48HCV 11656243 Ki > 630.96 nM T67162 CPE83G 11656848 Ki > 794.33 nM T67162 CT14BC 11657494 Ki = 1000 nM T67162 CP21DV 11658914 Ki = 120 nM T67162 C7NHO6 11659604 Ki = 64000 nM T67162 CD79UX 11661609 Ki = 150 nM T67162 CEL15N 11662194 Ki > 501.19 nM T67162 CE4FW0 11662306 Ki = 1 nM T67162 C6R1GA 11662426 Ki > 750 nM T67162 C4L7TV 11662592 Ki = 1.46 nM T67162 CBU0L8 11663504 Ki > 1000 nM T67162 C69RQX 11663526 Ki > 794.33 nM T67162 C3SJO5 11663578 Ki < 398.11 nM T67162 CO2HB4 11663604 Ki = 7.1 nM T67162 C1PB0O 11663999 Ki > 501.19 nM T67162 C16UWH 11664328 Ki > 794.33 nM T67162 CO69ZI 11666419 Ki > 10000 nM T67162 CPR2S8 11668034 Ki = 1500 nM T67162 CE34SW 11668495 Ki > 10000 nM T67162 C6URZ0 11668565 Ki = 2.5 nM T67162 CH82CY 11668731 Ki = 31.6 nM T67162 CNE2K5 11669953 Ki > 199.53 nM T67162 CY0J2U 11670421 Ki = 13 nM T67162 CQR15M 11670438 Ki > 1000 nM T67162 C2EUR0 11671211 Ki > 750 nM T67162 CGXE47 11672839 Ki = 7100 nM T67162 CH8M9X 11673558 Ki > 20000 nM T67162 CI26JH 11674133 Ki > 10000 nM T67162 CG01XN 11675208 Ki = 20.3 nM T67162 CDMZ42 11675785 Ki = 4.5 nM T67162 CH9M7J 11675867 IC50 = 6.6 nM T67162 CB4J2V 11675876 Ki = 730 nM T67162 CY4B9F 11676195 Ki = 16 nM T67162 C4KUL7 11676638 Ki = 53 nM T67162 CMQX39 11676873 Ki = 55.4 nM T67162 CWQ3M4 11677768 Ki < 398.11 nM T67162 CZ8XV7 11678072 Ki = 15 nM T67162 C6C4BJ 11678080 Ki > 630.96 nM T67162 CTK8R9 11678172 Ki = 28 nM T67162 CSQ4B1 11681599 Ki = 3.548 nM T67162 C6PW4M 11682536 Ki = 15 nM T67162 CVRW29 11682812 Ki = 280 nM T67162 C1ZD6V 11685267 Ki > 630.96 nM T67162 CS1WO0 11689612 Ki = 280 nM T67162 C7DLT5 11689690 Ki = 15.9 nM T67162 CRM26C 11691676 Ki > 1000 nM T67162 CG13YQ 11691697 Ki < 1000 nM T67162 C5J7PY 11692038 Ki > 750 nM T67162 CE1KI3 11692214 Ki > 1000 nM T67162 CGM36K 11692376 Ki = 630.96 nM T67162 C3LYZ6 11694483 Ki = 4000 nM T67162 CEQ6W7 11694810 Ki > 1000 nM T67162 C06BEA 11694873 Ki > 10000 nM T67162 CRO95K 11695189 Ki > 10000 nM T67162 C6R0CH 11696150 Ki = 1.778 nM T67162 CN1SJ8 11696598 Ki > 10000 nM T67162 C2G5DA 11696788 Ki = 4.3 nM T67162 CDV58J 11696813 Ki = 263 nM T67162 C1W8NR 11696910 Ki = 670 nM T67162 C9ED1Y 11697270 Ki = 28 nM T67162 CKT7L2 11698732 Ki = 2370 nM T67162 CT5J9M 11699340 Ki = 158.49 nM T67162 CB4H2O 11699469 Ki = 84 nM T67162 C2YE9V 11699516 Ki = 17 nM T67162 CFCB20 11699532 Ki < 316.23 nM T67162 CDLW51 11701907 Ki > 10000 nM T67162 CP0CH8 11704501 Ki = 4.7 nM T67162 CGD80W 11705119 Ki < 398.11 nM T67162 C2E8BF 11705395 Ki = 3.1 nM T67162 CLK68A 11705570 Ki > 630.96 nM T67162 CPC67X 11705929 Ki > 630.96 nM T67162 CJL61W 11706497 Ki = 140 nM T67162 C3EP0X 11708363 Ki > 20000 nM T67162 C0G1WQ 11709500 Ki > 10000 nM T67162 CPEA05 11710817 Ki = 11.4 nM T67162 CL08TQ 11711943 Ki = 9.6 nM T67162 CN8FE3 11712044 Ki > 630.96 nM T67162 CI3N1K 11716230 Ki > 10000 nM T67162 CZ6NB8 11716438 Ki = 19 nM T67162 CZ7SJ2 11716449 Ki = 82.6 nM T67162 C9FTL5 11718008 Ki = 2.5 nM T67162 CJH50P 11718173 Ki = 8.1 nM T67162 C7T1IL 11720119 Ki = 6.4 nM T67162 CGO56C 11720302 Ki = 35 nM T67162 CXUM63 11720838 Ki > 1000 nM T67162 C37DMH 11721190 Ki < 398.11 nM T67162 CS2H5V 11722531 Ki = 58.8 nM T67162 C2DMC4 11723696 Ki > 217 nM T67162 CCS8F5 11724853 Ki = 1100 nM T67162 C1N7MO 11725453 Ki = 498 nM T67162 CXYQ40 11725531 Ki = 44000 nM T67162 CNPU72 11725909 Ki = 330 nM T67162 CZLY39 11726130 Ki = 440 nM T67162 CRQ45H 11726532 IC50 = 13 nM T67162 CF7EC5 11729231 Ki = 3680 nM T67162 CVL96I 11729782 Ki = 47 nM T67162 C7UA6T 11730189 Ki = 71.9 nM T67162 C1JKS2 11731962 Ki = 13.54 nM T67162 CB8WF0 11732013 Ki = 571 nM T67162 C8L0KE 11732280 Ki = 81 nM T67162 C50XKE 11733317 Ki = 28.4 nM T67162 C2B7EY 11733372 Ki = 37 nM T67162 CP7IM3 11738945 EC50 > 10000 nM T67162 CB0T3F 11739255 Ki = 68.4 nM T67162 C9X7MJ 11739647 Ki > 1000 nM T67162 C43XLH 11739648 Ki > 1000 nM T67162 C5OR8S 11739823 EC50 > 10000 nM T67162 C0URA1 11740275 Ki = 316.23 nM T67162 CQP6N4 11743225 Ki = 7.943 nM T67162 CPG15O 11743399 IC50 > 1000 nM T67162 CYV02C 11747350 Ki = 59 nM T67162 C2J7KO 11751611 Ki > 10000 nM T67162 CG0YB2 11751828 Ki = 316.23 nM T67162 C5L2TO 11754850 Ki = 473 nM T67162 CD4Q5T 11761090 Ki = 48.7 nM T67162 C1MQ6G 11761374 Ki = 17.5 nM T67162 C5EH3J 11761412 EC50 = 1.7 nM T67162 CQX0T6 11762743 Ki = 512 nM T67162 C0KZ3P 11767026 Ki = 38.5 nM T67162 C0FM6J 11771801 Ki = 2530 nM T67162 CXS18C 11772112 Ki = 112 nM T67162 C1T7NR 11772242 Ki = 221 nM T67162 CVJN50 11772639 Ki > 1000 nM T67162 CXB48Q 11772767 Ki = 98.7 nM T67162 C9LUA7 11773414 Ki = 1700 nM T67162 C6T9RL 11773599 Ki = 20 nM T67162 CBI6Z0 11774041 EC50 > 10000 nM T67162 CV3OA5 11774865 Ki = 3.7 nM T67162 C5QGC3 11775544 Ki > 1000 nM T67162 CB46KD 11776309 EC50 > 10000 nM T67162 CN6BZ5 11777449 Ki = 614 nM T67162 CV91RG 11778580 Ki = 274 nM T67162 CK4IQ8 11778702 Ki = 134 nM T67162 C0L1XD 11779642 Ki = 640 nM T67162 C0CZ2S 11783381 Ki = 840 nM T67162 C3RAX7 11784937 Ki = 2110 nM T67162 C37LEP 11785183 Ki = 143 nM T67162 CT8LD5 11792163 Ki = 572 nM T67162 CAQP08 11792373 Ki = 5590 nM T67162 CE61JV 11793892 Ki = 1000 nM T67162 CAGO51 11793971 IC50 = 12 nM T67162 CHQ38Z 11794122 Ki = 4.8 nM T67162 CEW12K 11794570 Ki = 160 nM T67162 CU1EQ0 11794899 EC50 = 3.2 nM T67162 CJA41D 11795011 Ki = 3 nM T67162 CM82VH 11809382 Ki = 129 nM T67162 C19GOZ 11811640 Ki = 210 nM T67162 CN9M8E 11811722 IC50 = 538 nM T67162 CV68SD 11811808 Ki = 930 nM T67162 CWMA41 11812065 Ki = 120 nM T67162 CO5Y7T 11812299 Ki = 40 nM T67162 CGFW41 11812838 Ki = 414 nM T67162 CWFC60 11812905 Ki = 65.2 nM T67162 COB43E 11825520 Ki = 1100 nM T67162 C6IWM9 11826097 Ki = 20 nM T67162 CSNC92 11826347 Ki = 18 nM T67162 CJ1UD5 11826673 Ki = 36.79 nM T67162 CLR2Z9 11849181 Ki = 146 nM T67162 CLV61Z 11849182 Ki = 164 nM T67162 C0GM2D 11849184 EC50 > 10000 nM T67162 CL7YR2 11849225 EC50 > 10000 nM T67162 C37OPA 11849228 EC50 > 10000 nM T67162 CXG0L9 11849229 Ki = 140 nM T67162 C1HSM3 11849262 EC50 > 10000 nM T67162 CE83FP 11849263 EC50 > 10000 nM T67162 C5P7MQ 11849265 EC50 > 10000 nM T67162 C8X2RG 11849266 Ki = 60.9 nM T67162 CPXD54 11849267 Ki = 76.5 nM T67162 CPEZ08 11849268 Ki = 19.4 nM T67162 C9YEI0 11849298 EC50 > 10000 nM T67162 C78XQP 11849299 EC50 > 10000 nM T67162 CN8ST9 11849634 EC50 > 10000 nM T67162 CK80NX 11849635 EC50 > 10000 nM T67162 CFM1V9 11849684 EC50 > 10000 nM T67162 CKX4N9 11849729 EC50 > 10000 nM T67162 C0MNQ3 11849730 EC50 > 10000 nM T67162 CIG45B 11849731 EC50 > 10000 nM T67162 CD8B5E 11849734 EC50 > 10000 nM T67162 CJ5Y2T 11849735 EC50 > 10000 nM T67162 CEC2G8 11849736 Ki = 257 nM T67162 CO9E3X 11849774 EC50 > 10000 nM T67162 CU69CQ 11849775 Ki = 101 nM T67162 CXVA42 11849776 Ki = 125 nM T67162 CF6LX9 11849777 EC50 > 10000 nM T67162 C3URG4 11849778 Ki = 225 nM T67162 CY06BF 11849779 EC50 > 10000 nM T67162 CXA89H 11849780 EC50 > 10000 nM T67162 CG1H7P 11849781 EC50 > 10000 nM T67162 CZAX25 11849816 Ki = 25.3 nM T67162 C0XL3F 11849817 EC50 > 10000 nM T67162 C3D2KU 11849818 EC50 > 10000 nM T67162 CJ0N9Z 11849819 EC50 > 10000 nM T67162 CXY37C 11849820 EC50 = 366 nM T67162 CD8BQ7 11849821 Ki = 368 nM T67162 COWM39 11849822 EC50 > 10000 nM T67162 C4R6EA 11849823 EC50 > 10000 nM T67162 CUB53N 11857638 Ki = 55 nM T67162 C29HBR 11857639 Ki = 79 nM T67162 C29FMG 11857709 Ki = 83 nM T67162 CX50UR 11857710 Ki = 129 nM T67162 CW6V5E 11857711 Ki = 159 nM T67162 CD50HW 11857791 Ki = 23 nM T67162 CGL5D9 11857792 Ki = 69 nM T67162 CE0U9G 11857793 Ki = 37 nM T67162 CYJ5I7 11857794 Ki = 85 nM T67162 C9S5NU 11857861 Ki = 201 nM T67162 CU83FA 11857862 Ki = 88 nM T67162 CUO32E 11857863 Ki = 104 nM T67162 CD7O6J 11857864 Ki = 94 nM T67162 CXLW54 11948707 Ki = 2575 nM T67162 CK13QD 11953409 IC50 = 640 nM T67162 C23IVY 11957566 Ki = 1430 nM T67162 CPKV28 11957618 IC50 = 360 nM T67162 CNXB23 11957706 Ki = 310 nM T67162 C8JQL7 11957735 IC50 > 10000 nM T67162 C8IFT7 11973922 Ki = 5000 nM T67162 C9IH7R 11973925 Ki = 5000 nM T67162 CS7U5H 11973926 Ki = 5000 nM T67162 C7RY5S 11983282 EC50 = 1.7 nM T67162 CSFD67 11995339 Ki = 5000 nM T67162 CR4YS2 11996303 Ki = 158.49 nM T67162 C7D1AY 11996304 Ki = 31.62 nM T67162 CID7H8 12017581 Ki > 1000 nM T67162 C02JVQ 12049520 Ki = 1750 nM T67162 CXTH25 12049521 Ki = 330 nM T67162 C9V1XN 12049907 Ki = 1258.93 nM T67162 C1U7RH 12049908 Ki = 1258.93 nM T67162 C37GTL 12049910 Ki = 794.33 nM T67162 CVN2P5 12049911 Ki = 398.11 nM T67162 C57VXR 12050193 Ki = 440 nM T67162 CV56XD 12050194 Ki = 21500 nM T67162 C5C2GB 12050195 Ki = 790 nM T67162 C64JUP 12050196 Ki = 19500 nM T67162 C4QHA5 12050197 Ki = 85 nM T67162 CAL98J 12050198 Ki = 8650 nM T67162 CJ7W9T 12050199 Ki = 630 nM T67162 CXEV76 12050200 Ki = 13500 nM T67162 CP5W7X 12050201 Ki = 105 nM T67162 CZHQ31 12050202 Ki = 2000 nM T67162 CX47WZ 12052258 Ki = 15 nM T67162 C6QEW2 12066264 Ki = 379 nM T67162 CF4D5H 12066265 Ki = 625 nM T67162 C7NV4W 12068769 Ki > 10000 nM T67162 C9G7LR 12071089 Ki = 59 nM T67162 C4CE8D 12111141 Ki > 1500 nM T67162 CF4W7L 12269810 IC50 = 40 nM T67162 CRVU64 12280565 Ki = 1010 nM T67162 CT8SE7 12280575 Ki = 416 nM T67162 CHQ45V 12280580 Ki = 55.1 nM T67162 C4NWX9 12301195 Ki > 10000 nM T67162 CCLH20 12313091 Ki > 5000 nM T67162 C1QYW7 12461787 Ki = 13570 nM T67162 CS3JE5 12581154 Ki = 131 nM T67162 C9XLS6 12581156 Ki = 180 nM T67162 C72ZLP 12581164 Ki = 694 nM T67162 CU3XH9 12581203 Ki = 120 nM T67162 CEBK96 12581219 Ki = 181 nM T67162 C2CX7E 12668019 Ki = 8000 nM T67162 CK1X6Z 12741429 Ki = 3940 nM T67162 C5IVW7 12765116 Ki = 8.7 nM T67162 C28QEX 12765746 Ki = 1.1 nM T67162 C91ASK 12854846 Ki = 6309.57 nM T67162 CZT58X 12888943 Ki = 15 nM T67162 CNW1I4 12898419 Ki = 523 nM T67162 C8ON5D 12899499 Ki = 4.8 nM T67162 CY80HR 12899503 EC50 = 0.4 nM T67162 CPY6L8 12899569 Ki = 2.6 nM T67162 C6JX5B 12928483 Ki = 4408 nM T67162 CS3W4A 12937927 Ki > 217 nM T67162 C5MB7I 12997400 Ki = 3000 nM T67162 CXM15G 12997412 Ki = 473 nM T67162 CP0MN1 12997413 Ki = 1680 nM T67162 C9C2UY 13014680 Ki = 520 nM T67162 C1S2LW 13014681 Ki = 560 nM T67162 CG7T8B 13014683 Ki = 1400 nM T67162 CHI9P5 13014692 Ki = 1 nM T67162 C2V9FL 13091268 Ki = 0.309 nM T67162 C2VAE5 13091273 Ki = 2.3 nM T67162 CCG14E 13091356 Ki = 22 nM T67162 C1JW2Q 13091358 Ki = 22 nM T67162 CYN95Z 13091359 Ki = 2.9 nM T67162 C3BV2Q 13277350 Ki = 3.311 nM T67162 C0N7VC 13318472 Ki = 5 nM T67162 CC74ND 13373172 Ki = 486 nM T67162 CXLT95 13422623 Ki = 28 nM T67162 CB9J7Z 13493784 IC50 = 0.6761 nM T67162 CXYW07 13493789 IC50 = 5.248 nM T67162 C5TH3E 13493791 IC50 = 1.288 nM T67162 C4AG2Z 13493795 IC50 = 2.692 nM T67162 CI5Y6N 13611248 Ki > 10000 nM T67162 CJ75SB 13670706 Ki = 57 nM T67162 C86GDA 13680883 Ki > 100000 nM T67162 C39SGZ 13687192 Ki = 559 nM T67162 C3W2EN 13697621 Ki = 490 nM T67162 C3G8FK 13720686 EC50 = 174 nM T67162 C1EJ9C 13720688 EC50 = 137 nM T67162 C61ZDO 13720690 EC50 = 253 nM T67162 CP2I9Z 13720692 EC50 > 10000 nM T67162 C1CY0E 13720694 EC50 > 10000 nM T67162 C1H9QW 13767784 Ki = 652 nM T67162 C14SUX 13805900 Ki = 14 nM T67162 CN4Z2W 13851600 EC50 = 25 nM T67162 C1N5HM 13869506 Ki = 1050 nM T67162 CWS14H 13869641 Ki = 1.6 nM T67162 CSCP49 13869644 Ki = 7.762 nM T67162 C6E1DM 13922231 Ki = 826 nM T67162 CM40XI 13932579 Ki = 0.1549 nM T67162 CRH8V7 13994412 Ki = 551 nM T67162 CWL63T 14021682 IC50 = 3580 nM T67162 CYA3C2 14151052 Ki = 2.63 nM T67162 C50HOI 14198585 Ki = 19054.61 nM T67162 CIE29U 14198587 Ki = 144.54 nM T67162 CDE92A 14198590 Ki = 3715.35 nM T67162 CNYA85 14198594 Ki = 1819.7 nM T67162 COL2A4 14198597 Ki = 263.03 nM T67162 CTXB93 14198601 Ki = 1905.46 nM T67162 C5VD6K 14289494 Ki = 21 nM T67162 CV08GM 14378574 Ki = 113 nM T67162 C6E5IV 14576389 IC50 = 4.8 nM T67162 CSM29P 14665503 Ki = 0.85 nM T67162 CYW76P 14742527 Ki > 1000 nM T67162 CXZ7D8 14762911 IC50 = 8.318 nM T67162 CT19OL 14762912 IC50 = 45.71 nM T67162 CMO81H 14925759 Ki = 1096.48 nM T67162 CRE73S 14933735 Ki = 896 nM T67162 CTOY96 14944884 Ki = 153 nM T67162 C48XLF 14944887 Ki = 59 nM T67162 C47FIY 14950445 Ki = 857 nM T67162 C74OKN 14950446 Ki > 1667 nM T67162 C8RE3J 14950447 Ki = 215 nM T67162 CG96YX 14950448 Ki > 1000 nM T67162 CFS01M 14950449 Ki = 389 nM T67162 CY5P1M 14950450 Ki > 1000 nM T67162 C0VPR6 14950455 Ki = 44 nM T67162 CDT8C1 14950456 Ki > 333 nM T67162 CC47XA 14973078 Ki = 62 nM T67162 CY4E2W 14977566 Ki = 108 nM T67162 CZB32N 15006482 EC50 > 10000 nM T67162 C5MJ2V 15006484 EC50 > 10000 nM T67162 CDM02J 15006491 EC50 > 10000 nM T67162 CN0KL5 15021875 Ki = 204.17 nM T67162 C5F7NM 15021876 Ki = 104.71 nM T67162 C5W4MG 15034333 Ki > 10000 nM T67162 CL7P9W 15045455 Ki = 71 nM T67162 C4NG0F 15045457 EC50 = 4.9 nM T67162 CBQY50 15057516 IC50 = 5.1 nM T67162 C6ZUG1 15061351 IC50 = 420 nM T67162 C34UOH 15095973 IC50 = 3900 nM T67162 C3FKJ1 15111049 Ki = 5760 nM T67162 C2UD7Q 15111050 Ki = 629 nM T67162 CRE91W 15115512 Ki = 6.8 nM T67162 C4MD0E 15115513 Ki = 110 nM T67162 CR57HC 15115514 Ki = 4.8 nM T67162 CLX2W5 15115515 Ki = 7 nM T67162 CK59LT 15115516 Ki = 3.2 nM T67162 C8VT6W 15115519 Ki = 0.66 nM T67162 CV58UD 15115523 Ki = 1600 nM T67162 CGC27M 15115524 Ki > 5000 nM T67162 CHT4A5 15115525 Ki = 710 nM T67162 CBM63C 15124098 EC50 = 2 nM T67162 C1FGP8 15167693 IC50 = 67.61 nM T67162 C8N7IZ 15167695 IC50 = 257.04 nM T67162 COU62H 15167698 IC50 = 39.81 nM T67162 CE07GV 15167701 IC50 = 0.5012 nM T67162 CAF40B 15181802 IC50 = 41 nM T67162 CK46HZ 15225749 Ki = 647 nM T67162 CX8YP7 15229597 Ki = 131 nM T67162 CWJ2L5 15232472 Ki = 303 nM T67162 C5G3LK 15232474 Ki = 484 nM T67162 C36JOH 15232475 Ki = 1173 nM T67162 CNP2K1 15232476 Ki = 517 nM T67162 CV7ZG5 15232477 Ki = 703 nM T67162 C04JQR 15232482 Ki = 71 nM T67162 CUI42N 15291583 Ki = 56 nM T67162 C6CO3J 15291585 Ki = 6530 nM T67162 C76GUO 15291586 Ki = 3438 nM T67162 CQ30UI 15291587 Ki = 2345 nM T67162 C13GNK 15293841 Ki = 4250 nM T67162 C2XUE8 15344574 Ki = 374 nM T67162 CJIS26 15356306 Ki = 45.9 nM T67162 CH6A1U 15388745 Ki = 3.9 nM T67162 CDV47F 15389744 Ki = 7943.28 nM T67162 CGD3K7 15389746 Ki = 1862.09 nM T67162 CGZ5A0 15389747 Ki > 10000 nM T67162 C8US7F 15410404 Ki = 2.9 nM T67162 CFTI13 15410410 Ki = 0.47 nM T67162 CF6HQ7 15431693 Ki = 89 nM T67162 C4KNM7 15467369 Ki > 100000 nM T67162 C5UO3R 15467370 Ki = 48500 nM T67162 CCB94N 15467371 Ki = 7350 nM T67162 C2B0NM 15467372 Ki = 4000 nM T67162 CCMQ75 15467373 Ki = 8950 nM T67162 C5FWQ2 15508238 Ki = 8300 nM T67162 C8VB3H 15508239 Ki = 4900 nM T67162 C5NC6J 15508242 Ki = 49000 nM T67162 C72ERV 15512070 Ki = 1196 nM T67162 C30CHU 15512229 Ki < 316.23 nM T67162 CZ1L0V 15565706 IC50 = 52.48 nM T67162 CW50JX 15651970 Ki = 58882 nM T67162 CK5P6M 15651971 Ki = 3206 nM T67162 C59WZE 15654433 Ki = 48 nM T67162 CSD46O 15665503 Ki = 3.1 nM T67162 C98WHN 15665505 Ki = 255 nM T67162 CMK74C 15665506 Ki > 388 nM T67162 CU31EP 15665507 Ki = 58 nM T67162 CT6AY8 15665508 Ki = 1.8 nM T67162 CKQ42I 15665509 Ki = 5.7 nM T67162 C9SF4H 15665510 Ki = 5.8 nM T67162 CL2J4H 15665516 Ki = 41 nM T67162 C0NUO1 15665517 Ki = 2 nM T67162 CN94HR 15677951 Ki = 1040 nM T67162 CBXG85 15723715 Ki = 810000 nM T67162 CTPX97 15803947 Ki = 330 nM T67162 CUE15H 15817167 Ki = 865 nM T67162 CXG2S4 15817168 Ki = 293 nM T67162 C81RSY 15817169 Ki = 1403 nM T67162 CTPS81 15817172 Ki = 70 nM T67162 CT94FI 15817410 Ki = 1140 nM T67162 CD30XV 15840855 IC50 = 120 nM T67162 CW9M5X 15888352 Ki > 5000 nM T67162 C74UVA 15937765 Ki = 114 nM T67162 C0HAO3 15949564 Ki = 62.6 nM T67162 C8UO1X 15981509 Ki = 2500 nM T67162 C0G2EO 16007117 Ki = 181 nM T67162 C9CGE4 16007814 Ki = 300 nM T67162 CG4KC8 16038360 EC50 = 108 nM T67162 CT03WI 16040907 Ki = 390 nM T67162 CW5NS1 16041090 Ki = 288 nM T67162 C03VCW 16041091 Ki = 120 nM T67162 CM3O4Z 16041092 Ki = 54 nM T67162 CUL5M9 16041263 Ki = 33 nM T67162 C6S8AM 16041264 Ki = 84 nM T67162 CYTD80 16041265 Ki = 4.7 nM T67162 C86MYV 16041449 Ki = 6.5 nM T67162 CHF7K6 16041451 Ki = 1.2 nM T67162 CCJ65Y 16041628 Ki = 0.69 nM T67162 CE2Z7Y 16041629 Ki = 0.46 nM T67162 CRJX49 16041630 Ki = 2.4 nM T67162 CAUP23 16048564 Ki = 73 nM T67162 CCTM64 16049024 IC50 = 199.53 nM T67162 C17ZSM 16049026 IC50 = 794.33 nM T67162 CC3O5H 16049028 IC50 = 630.96 nM T67162 C71EWF 16049029 IC50 > 1000 nM T67162 C3OC9G 16049087 IC50 > 1000 nM T67162 CD41WM 16049088 IC50 > 1000 nM T67162 C63MIJ 16049090 IC50 = 3981.07 nM T67162 C8B4VS 16049158 IC50 = 2511.89 nM T67162 CE85LR 16049160 IC50 = 3981.07 nM T67162 C27VPK 16049162 IC50 = 501.19 nM T67162 C6Z4CS 16049234 IC50 = 1584.89 nM T67162 CP06JS 16049309 IC50 = 1000 nM T67162 CB3MN6 16049374 IC50 = 1584.89 nM T67162 C4QJE9 16049376 IC50 = 1000 nM T67162 C19EUK 16049377 IC50 = 3162.28 nM T67162 CKY42H 16049448 IC50 = 398.11 nM T67162 CC4F0L 16049450 IC50 > 794.33 nM T67162 C1SR0O 16071847 Ki > 5000 nM T67162 CWMC70 16090814 Ki = 1.5 nM T67162 CP09RQ 16090821 Ki = 38 nM T67162 CE61OV 16094664 Ki = 235 nM T67162 C5Q8DR 16094666 Ki = 127 nM T67162 C45TDZ 16094677 Ki > 10000 nM T67162 CTF8D7 16094681 Ki > 10000 nM T67162 CGA63F 16094698 Ki = 27 nM T67162 CH36CE 16094699 Ki = 3500 nM T67162 CZ1WJ4 16117151 Ki > 5000 nM T67162 CM32ZX 16117153 Ki > 5000 nM T67162 CXTB90 16117279 Ki > 5000 nM T67162 C1F2LS 16118795 Ki > 5000 nM T67162 C69VDS 16118923 Ki > 5000 nM T67162 CS1D0G 16121920 Ki = 2600 nM T67162 CYV05C 16123136 Ki = 251.19 nM T67162 C8C2IW 16123138 Ki = 63.1 nM T67162 C7YF8I 16123140 Ki = 100 nM T67162 C91DQN 16123241 Ki = 63.1 nM T67162 CQG7P8 16123247 Ki = 50.12 nM T67162 CA6D4S 16123347 Ki = 316.23 nM T67162 CBH5P4 16123349 Ki > 3162.28 nM T67162 CPN48R 16123353 Ki = 125.89 nM T67162 CK7H2W 16123462 Ki = 50.12 nM T67162 C5MY2Q 16123464 Ki = 1000 nM T67162 CNQ6J2 16123467 Ki > 3162.28 nM T67162 CJ4E9C 16277250 Ki > 7000 nM T67162 CZ2IS9 16660294 Ki > 10000 nM T67162 CGX0D5 16665071 Ki = 1.7 nM T67162 C2P0SB 16717791 EC50 > 10000 nM T67162 CHRG71 16738927 IC50 = 2511.89 nM T67162 CRIH69 16744003 Ki = 70 nM T67162 C3D0FE 16744004 Ki = 80 nM T67162 CKDM79 16744005 Ki = 400 nM T67162 CQ1MG0 16744171 Ki = 46 nM T67162 C1KNX9 16756402 Ki = 1400 nM T67162 CG35IB 16756405 Ki = 6100 nM T67162 CD2R9B 16756520 Ki = 780 nM T67162 CM9WO7 16756522 Ki = 1300 nM T67162 CM5CS7 16756524 Ki = 1000 nM T67162 CC6BN4 16756641 Ki = 120 nM T67162 C80KEV 16756642 Ki = 110 nM T67162 C5JZ4S 16756751 Ki = 1400 nM T67162 C4NC3P 16756752 Ki = 2900 nM T67162 CWF10J 16756753 Ki = 400 nM T67162 CTI89R 16759249 Ki = 68.1 nM T67162 C0LEG4 17159068 IC50 > 10000 nM T67162 CA6E9Q 17159204 IC50 > 10000 nM T67162 C8O7EW 17176477 IC50 = 4700 nM T67162 CHLR19 17424979 IC50 = 5100 nM T67162 C8ZK9L 17440212 IC50 = 7700 nM T67162 CF25CM 17449900 EC50 = 0.22 nM T67162 CH7C6A 17461770 Ki = 39.81 nM T67162 C73MFP 17469721 Ki = 6000 nM T67162 CPZJ30 17475863 Ki = 400 nM T67162 C3GD2P 17753379 Ki = 78 nM T67162 C7KP5T 17755866 Ki = 518 nM T67162 CX7VE8 17755867 Ki = 41.69 nM T67162 CUW8S4 17755868 Ki = 382 nM T67162 C3KA6Z 17755875 Ki > 10000 nM T67162 C4N1LS 17755991 Ki = 857 nM T67162 C6BE2Y 17755992 Ki > 10000 nM T67162 C10UQJ 17755999 Ki = 24.55 nM T67162 C6WO9X 17756101 Ki = 86.7 nM T67162 CI9RW0 17756102 Ki = 172 nM T67162 CDPT42 17756110 Ki > 10000 nM T67162 C0XG9B 17756212 Ki = 1396 nM T67162 C6JQ1K 17756213 Ki = 63 nM T67162 CTF31I 17866220 Ki = 251.19 nM T67162 CG69RD 17866221 Ki = 316.23 nM T67162 CR3A2X 17866228 Ki = 316.23 nM T67162 CZR2T6 17866229 Ki = 501.19 nM T67162 CV4N5L 17866237 Ki = 316.23 nM T67162 CP4YQ5 17866241 Ki = 398.11 nM T67162 C8D3RM 17866242 Ki = 398.11 nM T67162 C2ATF6 17866249 Ki = 316.23 nM T67162 CU9XT8 17867623 Ki = 79.43 nM T67162 CPQR14 17867626 Ki = 25.12 nM T67162 CL5C3X 17888044 IC50 = 81 nM T67162 C87POY 17895586 Ki = 100 nM T67162 C3HO5U 17895587 Ki = 125.89 nM T67162 CZ78BE 17987129 Ki > 1600 nM T67162 C9PV8A 18180076 IC50 > 10000 nM T67162 CMQT08 18397434 Ki = 3388.44 nM T67162 C9DQU7 18414156 Ki = 87.3 nM T67162 C94OZP 18427972 Ki = 74.13 nM T67162 CO8U1V 18613655 IC50 = 60 nM T67162 C23KVS 18649737 Ki = 12 nM T67162 CS5DZ1 18652674 Ki = 33.9 nM T67162 CW04FC 18702006 Ki = 79.43 nM T67162 CS5QC2 18702007 Ki = 25.12 nM T67162 CYI8L6 18702008 Ki = 39.81 nM T67162 CLK87H 18706871 Ki = 316.23 nM T67162 CGTJ59 18715674 Ki = 31.62 nM T67162 C3M6CU 18715682 Ki = 39.81 nM T67162 CPSI76 18797033 Ki = 199.53 nM T67162 C91OCW 18797049 Ki = 501.19 nM T67162 CVF4R7 18988817 Ki = 8.5 nM T67162 C08HLD 18988835 Ki = 11 nM T67162 CWXR15 18993044 Ki = 269 nM T67162 CW8PK0 19022852 Ki = 241 nM T67162 CREN73 19043055 Ki = 12.59 nM T67162 C0MY7J 19043056 Ki = 0.7943 nM T67162 C0MB8I 19370371 Ki = 808 nM T67162 C6AOE8 19426635 IC50 = 1698.24 nM T67162 CJ7RL6 19592091 Ki = 25.12 nM T67162 CT08UM 19592101 Ki = 316.23 nM T67162 C70DZN 19592119 Ki = 125.89 nM T67162 CG47ID 19592121 Ki = 125.89 nM T67162 C09EYA 19592126 Ki = 251.19 nM T67162 CO3QN2 19592133 Ki = 316.23 nM T67162 C8E3FM 19592141 Ki = 630.96 nM T67162 CMC12O 19592159 Ki = 100 nM T67162 CRF1H4 19608536 Ki = 3323 nM T67162 CW61QX 19694408 Ki = 199.53 nM T67162 CQN56J 19694436 Ki = 50.12 nM T67162 CCZ04S 19694443 Ki = 251.19 nM T67162 C10BRS 19694446 Ki = 31.62 nM T67162 CYJ3Z4 19694453 Ki = 316.23 nM T67162 C25YQI 19770958 IC50 > 10000 nM T67162 C1JTW4 19871273 Ki = 63.7 nM T67162 C61OBX 19881394 Ki = 1420 nM T67162 C43ACN 19938402 Ki = 4985 nM T67162 C1PS8O 19938405 Ki = 1414 nM T67162 CC8A3Z 19938408 Ki = 472 nM T67162 CEN3L5 19964401 Ki = 1300 nM T67162 C5IHG3 19964406 IC50 > 100000 nM T67162 C9VXS1 19964410 Ki = 400 nM T67162 CG5NT4 20035572 Ki > 10000 nM T67162 CG8Z4W 20256387 Ki > 300 nM T67162 C3DQS5 20267107 Ki > 3676 nM T67162 CB0NH7 20267108 Ki = 3676 nM T67162 C10IHJ 21073216 Ki = 1 nM T67162 CH8EN1 21073533 Ki = 2 nM T67162 C1R0SA 21073563 Ki = 2.5 nM T67162 CBUG29 21073579 Ki = 2.5 nM T67162 C15NJA 21073584 Ki = 1 nM T67162 CXMG13 21073587 Ki = 1 nM T67162 C57EJD 21073595 Ki = 5.7 nM T67162 CR0D3H 21073606 Ki = 1.6 nM T67162 C60WIT 21073656 Ki = 1 nM T67162 C6CQO1 21073658 Ki = 3 nM T67162 C1OL3G 21073667 Ki = 1.1 nM T67162 CVT16Y 21073690 Ki = 2 nM T67162 C9GHF5 21073716 Ki = 6 nM T67162 CA24ZJ 21073731 Ki = 1 nM T67162 CGP56E 21073788 Ki = 1 nM T67162 C6ARE1 21073793 Ki = 0.71 nM T67162 C3KMW4 21073817 Ki = 5 nM T67162 CHM64K 21073872 Ki = 2.6 nM T67162 C56JNM 21085427 Ki = 832 nM T67162 C9MDU4 21099413 Ki > 1000 nM T67162 CQU60A 21099448 Ki > 1000 nM T67162 CBCL34 21099463 Ki > 2000 nM T67162 C36INC 21099465 Ki > 1000 nM T67162 C6GRC9 21099470 Ki > 2000 nM T67162 CY75XP 21099472 Ki > 2000 nM T67162 CCO7D2 21099473 Ki > 2000 nM T67162 CDBY94 21099514 Ki > 1000 nM T67162 CB12UT 21099515 Ki > 1000 nM T67162 CP2R7D 21186098 IC50 = 250 nM T67162 CNR17B 21186102 IC50 = 50 nM T67162 CXY0P4 21186115 IC50 = 25 nM T67162 CY0QO4 21186124 IC50 = 23 nM T67162 C79MJX 21186138 IC50 = 60 nM T67162 CUJ4R9 21186143 IC50 = 490 nM T67162 CGY9F6 21186148 IC50 = 450 nM T67162 CRA23J 21186186 IC50 = 49 nM T67162 C18IWL 21186192 IC50 = 70 nM T67162 C5ER6Q 21186194 IC50 = 360 nM T67162 CLN86H 21219144 Ki = 1100 nM T67162 C2M0HK 21219154 Ki = 510 nM T67162 C1GQY9 21219156 Ki = 1200 nM T67162 C6LM2O 21219157 Ki = 6.1 nM T67162 C0W8PE 21219160 Ki = 460 nM T67162 CG4XF7 21219164 Ki = 370 nM T67162 C9S5XI 21219166 Ki = 450 nM T67162 CH83US 21219167 Ki = 1600 nM T67162 C60TBU 21219173 Ki > 1800 nM T67162 CB3KF6 21219176 Ki = 15 nM T67162 CPWG76 21302447 Ki = 16 nM T67162 CQF01H 21302453 Ki = 14 nM T67162 CTFH75 21302454 Ki = 4.7 nM T67162 CGL9D3 21302455 Ki = 2.3 nM T67162 CY3M2Z 21302456 Ki = 50 nM T67162 CY6H3F 21302457 Ki = 15 nM T67162 CB4V8Q 21302458 Ki = 6 nM T67162 C9WD5O 21302459 Ki = 31 nM T67162 C7TSU2 21302471 Ki = 4.7 nM T67162 CJ30ZL 21345773 Ki = 300 nM T67162 CHN7Y1 21390740 Ki = 131.83 nM T67162 C94BPG 21460314 Ki = 262 nM T67162 C7MYT1 21462964 Ki = 1100 nM T67162 C8GC6E 21462980 Ki = 640 nM T67162 C2D6ZX 21465540 Ki > 1700 nM T67162 C3T5HF 21509921 Ki = 831.76 nM T67162 CFN81Q 21527771 Ki = 1.072 nM T67162 CH59WN 21533446 Ki = 2.089 nM T67162 CL5A2V 21554999 Ki > 10000 nM T67162 C61LUT 21555004 Ki > 10000 nM T67162 C4B0TN 21557475 Ki = 1302 nM T67162 CRE80D 21559988 Ki = 470 nM T67162 CZLT46 21559989 Ki = 1.905 nM T67162 CAH39X 21564536 Ki > 10000 nM T67162 C0IQ2X 21604779 IC50 = 8.71 nM T67162 CVF4N8 21786101 EC50 = 0.65 nM T67162 CT7XG9 21830793 Ki > 10000 nM T67162 CXJG29 21852778 EC50 = 1913 nM T67162 CG08FZ 21969199 Ki = 501.19 nM T67162 C0EGL8 21969201 Ki = 63.1 nM T67162 C4TQ5H 21969204 Ki = 316.23 nM T67162 C20AOH 21969205 Ki = 501.19 nM T67162 CMH48V 21973550 Ki = 199.53 nM T67162 CW90QB 21997225 Ki = 185 nM T67162 CSQ2Y0 22017550 Ki > 1000 nM T67162 CLF09T 22065962 Ki = 1170 nM T67162 C5FS6A 22082742 Ki > 5000 nM T67162 CYCS06 22100932 Ki = 2000 nM T67162 CM75DA 22100933 Ki = 590 nM T67162 CP48JW 22100940 Ki = 600 nM T67162 C68MQE 22100943 Ki = 340 nM T67162 CWH1R0 22100957 Ki > 1700 nM T67162 C9TG8S 22100962 Ki > 1600 nM T67162 CLCN93 22100964 Ki > 1800 nM T67162 CC3LF7 22100965 Ki > 2000 nM T67162 C90FER 22100968 Ki = 240 nM T67162 C9RUA4 22100970 Ki = 670 nM T67162 C4SXJ3 22132503 Ki = 630.96 nM T67162 CS62AZ 22261332 Ki = 19.3 nM T67162 C2M4SX 22261340 Ki = 7.37 nM T67162 C0FTG5 22376257 Ki = 125.89 nM T67162 CKL08Z 22397822 Ki = 251.19 nM T67162 C5ER0Q 22397830 Ki = 180 nM T67162 C9U1GM 22403029 Ki = 7.943 nM T67162 CGVE83 22403039 Ki = 7.943 nM T67162 C9KI2W 22403044 Ki = 251.19 nM T67162 C3FEL1 22403055 Ki = 316.23 nM T67162 CUNF84 22403068 Ki = 158.49 nM T67162 CM6YV2 22403070 Ki = 1.995 nM T67162 CY0ZF7 22403109 Ki = 158.49 nM T67162 CCZ3U1 22403110 Ki = 398.11 nM T67162 C3GWZ7 22403137 Ki = 0.7943 nM T67162 CCZ5Q3 22622605 Ki = 25.12 nM T67162 CVX19H 22727322 Ki = 3388 nM T67162 CT45YC 22727323 Ki = 295 nM T67162 CL26HS 22727324 Ki = 321 nM T67162 CCS83F 22727331 Ki = 440 nM T67162 CS5J2U 22727332 Ki = 585 nM T67162 CAUK40 22727334 Ki = 3366 nM T67162 CSCJ35 22727335 Ki = 1727 nM T67162 CCIW17 22727346 Ki = 1401 nM T67162 CS9IF2 22727347 Ki = 964 nM T67162 CFQ92N 22727351 Ki = 1470 nM T67162 CE2P3H 22727356 Ki = 9724 nM T67162 C64UKQ 22727358 Ki = 4136 nM T67162 CU6B2Z 22727361 Ki = 2196 nM T67162 C5WCD3 22745278 IC50 > 10000 nM T67162 CA02UK 22849991 Ki = 3.1 nM T67162 C5DJR8 22849992 Ki = 3.6 nM T67162 C4S2NC 22876327 Ki = 19.95 nM T67162 CAM3H4 22910005 Ki = 9.7 nM T67162 C04FIU 22953120 Ki = 183 nM T67162 C8C3VU 23025506 Ki > 100000 nM T67162 C8IN9H 23202795 Ki = 12.59 nM T67162 C16PUX 23202799 Ki = 100 nM T67162 CVAB38 23202826 Ki = 15.85 nM T67162 CH5C7X 23288790 Ki = 348 nM T67162 CP41OK 23322039 EC50 = 85 nM T67162 CLME84 23363843 Ki = 1225 nM T67162 CEP65L 23364995 Ki = 4.5 nM T67162 CD78OT 23424166 Ki = 32.36 nM T67162 CQSF94 23625084 Ki = 78 nM T67162 CNAK80 23625241 Ki = 83 nM T67162 CVRW14 23625242 Ki = 125 nM T67162 C4K8QX 23625243 Ki = 47 nM T67162 CPR07Q 23625244 Ki = 149 nM T67162 C43MPJ 23625385 Ki = 111 nM T67162 CRB85L 23625386 Ki = 560 nM T67162 CS0VM3 23625539 Ki = 44 nM T67162 CD7AK1 23625540 Ki = 78 nM T67162 C85WQO 23625541 Ki = 49 nM T67162 CESF95 23625542 Ki = 68 nM T67162 C9Z1EM 23625543 Ki = 52 nM T67162 CU0F6C 23625706 Ki = 159 nM T67162 CXD3E6 23625925 Ki = 112.2 nM T67162 CK6B7G 23630497 Ki = 251.19 nM T67162 CH95VG 23630499 Ki = 316.23 nM T67162 C2XLN1 23630501 Ki = 501.19 nM T67162 C1N5TV 23630503 Ki > 1258.93 nM T67162 C7WZJ0 23630505 Ki = 630.96 nM T67162 C4MI9Y 23630602 Ki = 125.89 nM T67162 C24TDZ 23630604 Ki = 79.43 nM T67162 CU8D0O 23630606 Ki = 199.53 nM T67162 CKB1E5 23630796 Ki > 794.33 nM T67162 CJ81PU 23630797 Ki = 251.19 nM T67162 CV68XN 23630900 Ki = 630.96 nM T67162 CD61SO 23630901 Ki = 1258.93 nM T67162 CY2RG1 23630902 Ki = 1000 nM T67162 CJ90YG 23630903 Ki = 1995.26 nM T67162 CTJS17 23630998 Ki = 6309.57 nM T67162 CXVR30 23630999 Ki = 398.11 nM T67162 CSAT45 23631000 Ki = 501.19 nM T67162 C6EO1W 23631001 Ki > 1584.89 nM T67162 CE3AM4 23631091 Ki > 398.11 nM T67162 C9BMW2 23631092 Ki = 199.53 nM T67162 CKT7B3 23631093 Ki = 158.49 nM T67162 CM8U1D 23631172 Ki = 1258.93 nM T67162 CWZT34 23631173 Ki = 7.943 nM T67162 CH2I1P 23631366 Ki = 398.11 nM T67162 C6YS4P 23631368 Ki = 1000 nM T67162 C4TV8X 23631454 Ki = 398.11 nM T67162 CE40PT 23631458 Ki = 158.49 nM T67162 C09NTA 23631540 Ki = 251.19 nM T67162 C83QKW 23631544 Ki = 1258.93 nM T67162 C0RPW8 23631636 Ki = 1000 nM T67162 CI4B6N 23642427 Ki = 0.68 nM T67162 CPZV02 23643663 Ki = 15 nM T67162 CX93TK 23643870 Ki = 32 nM T67162 CO4C6M 23653115 Ki = 1.2 nM T67162 CBUJ02 23653176 Ki = 375 nM T67162 CA8ZX6 23731422 Ki = 17.78 nM T67162 C2BO0F 23928184 Ki = 275 nM T67162 C8X0BG 23964891 Ki > 42000 nM T67162 CDH38J 23992579 Ki = 2179 nM T67162 CQ0KU9 24738459 Ki = 3.18 nM T67162 C3RS6J 24742011 EC50 = 2.22 nM T67162 C7BCW8 24754330 Ki = 638 nM T67162 C9SP0R 24754332 Ki = 90.6 nM T67162 C20IKD 24754400 EC50 = 1.56 nM T67162 CP0VE5 24754476 Ki = 14.6 nM T67162 CFEP49 24754538 Ki = 167 nM T67162 C5GYO8 24754540 Ki = 21.7 nM T67162 CYGH43 24754542 Ki = 26 nM T67162 C2XAQ7 24754913 Ki = 649 nM T67162 C39ZCR 24754914 Ki = 24.6 nM T67162 CWA40O 24754983 Ki = 70.3 nM T67162 CJ1QB7 24758481 Ki = 398.11 nM T67162 C8CWX4 24758715 Ki = 39.81 nM T67162 CU06GI 24758717 Ki = 251.19 nM T67162 CPL05Y 24758828 Ki = 501.19 nM T67162 C7RZ9I 24758830 Ki = 316.23 nM T67162 C6JQC4 24758832 Ki = 251.19 nM T67162 CBNF87 24758834 Ki = 1000 nM T67162 CGQL10 24758836 Ki = 398.11 nM T67162 CGE32Q 24758838 Ki > 3162.28 nM T67162 CL80CU 24758945 Ki = 398.11 nM T67162 C8JQW6 24758947 Ki = 316.23 nM T67162 CMB3J9 24759792 EC50 = 269.15 nM T67162 C6B1IG 24767784 Ki = 1.2 nM T67162 C6Z1PX 24768516 Ki = 173 nM T67162 C0HO5Q 24768517 Ki = 123 nM T67162 CX7E3K 24768518 Ki = 60 nM T67162 CW3PD4 24768519 Ki > 1000 nM T67162 C9G8ZH 24768520 Ki = 107 nM T67162 C9UOG8 24768522 Ki > 1000 nM T67162 CS8YX3 24768523 Ki > 1000 nM T67162 CSW50R 24768524 Ki = 292 nM T67162 CW8N2E 24768525 Ki > 1000 nM T67162 C0I2HU 24769156 Ki > 1000 nM T67162 CD7CV6 24771120 Ki > 2000 nM T67162 CP08DV 24805120 Ki = 501.19 nM T67162 CI15OJ 24805284 Ki = 1202.26 nM T67162 C21VNW 24805285 Ki = 776.25 nM T67162 CKW7R2 24805286 Ki = 1479.11 nM T67162 CQ7S8N 24805287 Ki = 2041.74 nM T67162 C9K0CX 24805674 Ki = 5.6 nM T67162 C8TZY0 24810004 Ki = 132 nM T67162 CSCW01 24815434 Ki = 25.12 nM T67162 CBF6J9 24815439 Ki = 39.81 nM T67162 C0DYP7 24815883 Ki = 125.89 nM T67162 CN9AY0 24815976 Ki = 251.19 nM T67162 CYL30C 24823920 Ki = 220 nM T67162 CHC2B6 24823921 Ki = 150 nM T67162 C0Y8UL 24823922 Ki = 150 nM T67162 CB9Z8R 24824060 Ki = 1700 nM T67162 CTS57E 24824061 Ki = 550 nM T67162 C6ED9B 24824062 Ki = 46 nM T67162 CPT34W 24824063 Ki = 30000 nM T67162 CGU94D 24824065 Ki = 4500 nM T67162 C6Y4FV 24824066 Ki = 6100 nM T67162 C58AMS 24829343 Ki = 950 nM T67162 C1OFA6 24837531 IC50 = 1530 nM T67162 CDC91N 24839550 Ki < 10000 nM T67162 CF8I9P 24845776 Ki = 1000 nM T67162 C2T5EW 24847750 IC50 > 0.00001 nM T67162 C2A0LT 24849462 Ki = 15.85 nM T67162 CUW23K 24854106 Ki = 330 nM T67162 C2OM6C 24863698 Ki = 389.05 nM T67162 CO51AG 24863961 Ki > 10000 nM T67162 CD9SF2 24863962 Ki > 10000 nM T67162 C3HK0J 24865725 Ki = 63.1 nM T67162 C0O6FX 24865727 Ki = 501.19 nM T67162 CBGO31 24867245 Ki = 279 nM T67162 C1FZV4 24873453 Ki = 703 nM T67162 CKG9N0 24873454 Ki = 2288 nM T67162 CKF9G6 24878061 Ki = 6800 nM T67162 CV1PY2 24878951 Ki > 10000 nM T67162 CK6JC4 24878953 Ki = 266 nM T67162 C4SL0V 24879001 Ki = 213 nM T67162 C3Z4JN 24879003 Ki > 10000 nM T67162 C56IDA 24879005 Ki > 10000 nM T67162 C23LNY 24879008 Ki = 516 nM T67162 C9C8OH 24879010 Ki = 146 nM T67162 C1ZRH6 24879054 Ki > 10000 nM T67162 CD17RE 24879056 Ki > 10000 nM T67162 CX20BZ 24879058 Ki > 10000 nM T67162 C43RTZ 24882193 IC50 = 700 nM T67162 C98ZIV 24882509 IC50 = 1000 nM T67162 C49GLI 24882561 Ki = 760 nM T67162 CI53SE 24893978 Ki = 100 nM T67162 CAOF91 24894071 IC50 > 10000 nM T67162 C3C0KP 24894134 EC50 > 50000 nM T67162 C13JLE 24900426 IC50 = 316.23 nM T67162 C69AYD 24900557 Ki = 48.98 nM T67162 C1U9VL 24900685 IC50 = 1584.89 nM T67162 CU3F7K 24900689 EC50 = 251.19 nM T67162 CPLO51 24900749 IC50 = 1000 nM T67162 CX69CF 24900750 IC50 = 794.33 nM T67162 CE5W9U 24900751 IC50 = 1258.93 nM T67162 CQDR84 24900811 IC50 = 2511.89 nM T67162 CIL8Q7 24900812 IC50 = 5011.87 nM T67162 C9YUP8 24900813 IC50 = 630.96 nM T67162 C63ILV 24900872 IC50 > 2511.89 nM T67162 CSF3J2 24900874 IC50 > 10000 nM T67162 C4AT0P 24900937 IC50 = 3162.28 nM T67162 C2NR7M 24900942 IC50 = 1000 nM T67162 CW0QV2 24901141 IC50 = 251.19 nM T67162 CHWE43 24901143 IC50 = 251.19 nM T67162 C5ZCX4 24901144 IC50 = 398.11 nM T67162 CNP40V 24901209 IC50 = 398.11 nM T67162 C7MGC9 24901210 IC50 = 630.96 nM T67162 CS6BH7 24901211 IC50 > 794.33 nM T67162 C4JB7G 24901283 IC50 = 794.33 nM T67162 CBS0V5 24901284 IC50 = 79.43 nM T67162 C83MAF 24901285 IC50 = 125.89 nM T67162 CVE24O 24901347 IC50 = 1995.26 nM T67162 CV5GY0 24901348 IC50 = 1000 nM T67162 CFZ5D7 24901349 IC50 = 1995.26 nM T67162 CCMQ16 24901351 IC50 = 630.96 nM T67162 CGW2U6 24901413 IC50 > 794.33 nM T67162 COY5H0 24901416 IC50 = 794.33 nM T67162 C4IGH9 24936042 Ki = 14 nM T67162 CAP8R4 24936081 EC50 = 19.9 nM T67162 C5MYC3 25010776 IC50 = 4500 nM T67162 C6DO4B 25032525 Ki = 15 nM T67162 CYJ5G1 25067564 Ki = 2910 nM T67162 C7O8YH 25068794 Ki = 34 nM T67162 CZ9SN8 25068797 Ki = 24.7 nM T67162 CL46IP 25068850 Ki = 40.7 nM T67162 CEH7D9 25068903 Ki = 80.7 nM T67162 CB03DL 25068905 Ki = 16.3 nM T67162 C5ZHN9 25068906 Ki = 27.8 nM T67162 C0ZJB7 25068907 Ki = 13.6 nM T67162 C9G7EM 25068908 Ki = 44.5 nM T67162 CZBY61 25068962 Ki = 290 nM T67162 CP9G5Z 25068963 Ki = 2.63 nM T67162 CB3F0I 25068964 Ki = 0.302 nM T67162 CCO7B3 25068966 Ki = 12.1 nM T67162 C16ERI 25069015 Ki = 10.2 nM T67162 CZM94A 25069016 Ki = 4.47 nM T67162 CYZ45N 25069072 Ki = 11.48 nM T67162 CEB96S 25069073 Ki = 1.54 nM T67162 CAI7V1 25069074 Ki = 22.3 nM T67162 C8A3HM 25069121 Ki = 0.0575 nM T67162 CG5WX6 25069122 Ki = 0.575 nM T67162 CS8VK1 25069125 Ki = 2.08 nM T67162 CHZB81 25069180 Ki = 8.23 nM T67162 C3W1AX 25069181 Ki = 0.5754 nM T67162 CPGZ03 25069239 Ki = 8.92 nM T67162 CT0R3H 25069240 Ki = 5.81 nM T67162 CX5JF4 25069241 Ki = 9.54 nM T67162 C1P4EC 25069242 Ki = 1.86 nM T67162 CCV27I 25069243 Ki = 0.877 nM T67162 C5BR0K 25069297 Ki = 11.2 nM T67162 CU34CX 25069298 Ki = 1.41 nM T67162 C0Z6YL 25069299 Ki = 0.891 nM T67162 C5Z9MA 25069300 Ki = 13.8 nM T67162 C1OGS2 25069301 Ki = 10.3 nM T67162 C53LJG 25069302 Ki = 5.49 nM T67162 CX74UK 25069353 Ki = 8.59 nM T67162 C8F6VC 25069354 Ki = 22.3 nM T67162 C56RCY 25069355 Ki = 5.75 nM T67162 CI7SM5 25069356 Ki = 15.8 nM T67162 CD0YW2 25070416 Ki = 10 nM T67162 C5QU0F 25070419 Ki = 9.4 nM T67162 CTN36E 25070740 Ki = 25 nM T67162 CGAZ01 25070742 Ki = 24 nM T67162 CKB23A 25071066 Ki = 34 nM T67162 CI8NL3 25071384 Ki = 3.2 nM T67162 C6F5SU 25071385 Ki = 1.8 nM T67162 CL7TN4 25071691 Ki = 0.17 nM T67162 C75ZIC 25071692 Ki = 0.32 nM T67162 C49ZFU 25072002 Ki = 0.16 nM T67162 CM28GQ 25072632 Ki = 2.1 nM T67162 C8OBV4 25072633 Ki = 0.74 nM T67162 CIT6G4 25072635 Ki = 6.2 nM T67162 CS1CI4 25072941 EC50 = 2.6 nM T67162 C3CLH5 25072943 Ki = 16 nM T67162 C1XSD0 25072946 Ki = 15 nM T67162 CBKG34 25093832 Ki = 0.094 nM T67162 C3W6DQ 25096873 Ki = 0.81 nM T67162 C2YJX3 25099159 Ki = 213.8 nM T67162 CXA09P 25107515 Ki = 40 nM T67162 CDW7J5 25107516 Ki = 1.3 nM T67162 C81QKN 25107517 Ki = 22 nM T67162 C1QE6A 25107519 Ki = 226 nM T67162 C3VY8O 25107520 Ki = 185 nM T67162 CYE53P 25107578 Ki = 21 nM T67162 CJO1X8 25107579 Ki = 5.3 nM T67162 C59IVO 25107580 Ki = 20 nM T67162 CMPG74 25107581 Ki = 30 nM T67162 CNW7A8 25107582 Ki = 7.8 nM T67162 CU71RN 25107583 Ki = 91 nM T67162 C8ZM2J 25107647 Ki = 93 nM T67162 CJF71U 25107648 Ki = 362 nM T67162 C6M9LD 25107649 Ki = 33 nM T67162 CEM90Y 25107650 Ki = 9.2 nM T67162 C2JW3O 25107651 Ki = 64 nM T67162 C7M1XT 25107652 Ki = 501 nM T67162 C4ASH8 25107717 Ki = 311 nM T67162 CQ71NR 25107718 Ki = 723 nM T67162 C3NGR5 25108474 Ki = 96 nM T67162 C8GW4P 25108475 Ki = 65 nM T67162 CJK06X 25110705 Ki = 29 nM T67162 CVIB80 25110709 Ki = 210 nM T67162 C50IKG 25110765 IC50 > 10000 nM T67162 C9DZN4 25128753 Ki = 225 nM T67162 CT7U5K 25128755 Ki = 554 nM T67162 C2FY7C 25128757 Ki = 12.9 nM T67162 CPZ7K5 25128759 Ki = 280 nM T67162 CL1HC0 25129111 Ki = 1.7 nM T67162 C8MX9U 25129113 Ki = 4.9 nM T67162 C2U0HS 25129115 Ki = 1.5 nM T67162 C0I8HD 25129458 Ki = 5.6 nM T67162 CTX43Q 25129459 Ki = 1.5 nM T67162 C6XMF9 25129460 Ki = 11.7 nM T67162 C5NW4M 25129807 Ki = 33.4 nM T67162 C2O4KV 25129809 Ki = 41.4 nM T67162 CQKP18 25130148 Ki = 41.69 nM T67162 CX3R5L 25130151 Ki = 565 nM T67162 CD2KY1 25130153 Ki = 39.4 nM T67162 C3I1FU 25130155 Ki = 29.8 nM T67162 CAV81B 25130157 Ki = 1.06 nM T67162 CRSZ60 25130159 Ki = 40.1 nM T67162 C7TQ4B 25130505 Ki > 10000 nM T67162 CIM1F4 25130509 Ki = 1.4 nM T67162 CD04PQ 25130829 Ki = 85.11 nM T67162 CM58BO 25130830 Ki = 12.02 nM T67162 C9HYT3 25130831 Ki > 10000 nM T67162 C36NMK 25130836 Ki = 15.85 nM T67162 C1MNU0 25131483 Ki > 10000 nM T67162 CZ6NK0 25131829 Ki > 10000 nM T67162 CFJ6Y9 25131876 Ki = 12.3 nM T67162 C67QCG 25132869 Ki = 35.3 nM T67162 CC0S6N 25132870 Ki = 545 nM T67162 CG9I6X 25132871 Ki = 196 nM T67162 C8Y5LD 25133211 Ki = 2070 nM T67162 CGBL04 25139014 Ki > 10000 nM T67162 CN61ZL 25139180 Ki = 4700 nM T67162 CLTF40 25139181 Ki = 40 nM T67162 CN32VX 25139329 Ki = 180 nM T67162 C0LZ7B 25139335 Ki = 2100 nM T67162 CW07GC 25139477 Ki = 220 nM T67162 CQD6N1 25139478 Ki = 670 nM T67162 CN3S7R 25139479 Ki = 170 nM T67162 CSG25V 25139481 Ki = 4700 nM T67162 CJ5VX0 25140466 Ki = 6280 nM T67162 CXDM41 25141533 Ki = 249 nM T67162 CL84YJ 25141534 EC50 = 170 nM T67162 CX04LB 25142456 Ki = 1910 nM T67162 CW2PL7 25155850 Ki = 298000 nM T67162 C4UXF6 25155851 Ki > 1000000 nM T67162 C65LWZ 25156129 Ki = 1412000 nM T67162 CS3Q4N 25156130 Ki = 427000 nM T67162 CZ04VO 25156131 Ki = 6300 nM T67162 C6MXE3 25156132 Ki > 1000000 nM T67162 CU5C7V 25156133 Ki = 655000 nM T67162 C65FNY 25156411 Ki = 847000 nM T67162 CKIH98 25156412 Ki = 629000 nM T67162 C35NHX 25156413 Ki = 854000 nM T67162 C94OIG 25156414 Ki = 565000 nM T67162 C1IEF6 25156415 Ki > 1000000 nM T67162 CL1B2G 25156416 Ki = 114000 nM T67162 CUX0F4 25156684 Ki > 1000000 nM T67162 CB4A2S 25156685 Ki > 1000000 nM T67162 CJO48V 25156686 Ki > 1000000 nM T67162 CF27EQ 25156688 Ki > 1000000 nM T67162 C8U6PV 25156966 Ki > 1000000 nM T67162 C05TOB 25157253 Ki = 1324000 nM T67162 CYM3H9 25157257 Ki = 20000 nM T67162 CS0E3J 25157260 Ki = 178000 nM T67162 CQI4S2 25157543 Ki > 1000000 nM T67162 C6Y4AJ 25157546 Ki > 1000000 nM T67162 CKP10W 25157549 Ki > 1000000 nM T67162 C9B0UR 25157845 Ki > 1000000 nM T67162 CX2CP8 25157848 Ki > 1000000 nM T67162 C1XP3Q 25157850 Ki > 1000000 nM T67162 C5J4ES 25158433 Ki > 1000000 nM T67162 COK46A 25158434 Ki > 1000000 nM T67162 CQRL83 25158435 Ki = 67000 nM T67162 C26IMW 25158436 Ki > 1000000 nM T67162 C78HME 25212275 Ki = 47 nM T67162 CE6Z9I 25212276 Ki = 146 nM T67162 CJ1Z9H 25216680 Ki > 10000 nM T67162 C1T3LR 25218143 Ki > 10000 nM T67162 CPI03N 25218397 Ki > 10000 nM T67162 CL1R3Q 25218401 Ki > 10000 nM T67162 COV83Z 25256814 Ki = 7 nM T67162 C76ROY 25256815 Ki = 35.48 nM T67162 C7JZ2D 25256816 Ki = 1.5 nM T67162 C6PL1Y 25256817 Ki = 36.31 nM T67162 CM2T9Y 25263297 Ki > 2000 nM T67162 CFJM71 25263302 Ki > 2000 nM T67162 C2QLS7 25375331 Ki = 5698 nM T67162 CRB9W7 25450664 Ki > 10000 nM T67162 C8FWE5 25456694 Ki = 6787 nM T67162 CEK31Q 25487292 Ki > 10000 nM T67162 CN39GC 25491778 Ki > 10000 nM T67162 CSW0O8 25895957 Ki > 1000 nM T67162 CPD3L4 25895959 Ki = 450 nM T67162 CR89HN 27039365 Ki = 180375 nM T67162 C4MRQ0 27842480 EC50 > 10000 nM T67162 CUP73X 27846388 IC50 = 9000 nM T67162 C0BJ5F 27846916 IC50 = 535 nM T67162 CYG87R 27847327 IC50 > 10000 nM T67162 C1QT2Y 28071610 Ki > 10000 nM T67162 CU9PY2 28357663 Ki = 2233 nM T67162 CYKH58 28390601 Ki = 1245 nM T67162 C6RQ4D 29945476 EC50 = 1496 nM T67162 CE0PR6 30616772 Ki = 8053 nM T67162 CAB4L3 30740059 Ki = 59 nM T67162 CM12QP 30743524 Ki = 5847 nM T67162 CDY01I 30982708 Ki = 4.8 nM T67162 C9R0CK 31281277 IC50 > 100000 nM T67162 CB59EX 31343434 EC50 > 100000 nM T67162 CEZ1A6 32718395 Ki = 3195 nM T67162 C9QGK3 34257212 Ki > 1000 nM T67162 CFE27P 35995182 EC50 = 3500 nM T67162 C8VRX4 36717024 EC50 > 50000 nM T67162 CX8IT3 38417721 EC50 = 5200 nM T67162 C20XSK 39729535 EC50 = 24000 nM T67162 C15PLV 40152769 Ki = 60 nM T67162 C8R2PE 40517075 Ki = 6700 nM T67162 CY1O0S 41532205 Ki = 37 nM T67162 CDP76A 42266865 Ki = 890 nM T67162 C2NS9O 42266974 Ki = 2511.89 nM T67162 CG2KD8 42273483 Ki < 10000 nM T67162 CG56DF 42388639 Ki = 132 nM T67162 C0XMS9 42605994 Ki = 73000 nM T67162 CD61JW 42606339 Ki = 20000 nM T67162 C0TN5O 42606573 Ki = 27000 nM T67162 CDE4U8 42609932 Ki = 5.92 nM T67162 CAM63X 42618195 IC50 > 1000 nM T67162 C8K4UF 42618197 IC50 > 1000 nM T67162 CK3QD2 42625354 Ki = 60 nM T67162 C0P3JR 42626172 Ki = 217 nM T67162 CZ19KX 42626240 Ki = 715 nM T67162 CTL2I7 42626243 Ki = 328 nM T67162 CLH7Y0 42626289 Ki = 34 nM T67162 C5VTZ6 42626293 Ki = 153 nM T67162 CRQ91B 42626318 Ki = 295 nM T67162 CY7W2J 42631003 Ki = 85.11 nM T67162 C0AI7N 43229249 Ki = 645.65 nM T67162 C75LHU 43398192 Ki > 30000 nM T67162 CEL6J0 44123782 Ki = 62 nM T67162 C03RGW 44182375 Ki = 150 nM T67162 C2AV1K 44190762 IC50 = 3550 nM T67162 C6SG0O 44192200 Ki = 1306 nM T67162 CS4TB9 44203057 Ki = 5.2 nM T67162 CMR7T1 44204999 Ki = 0.5012 nM T67162 CVG6X1 44209472 Ki = 186 nM T67162 CD5AB7 44209480 Ki = 124 nM T67162 CBA7V5 44212307 Ki = 100 nM T67162 CM76LY 44212310 Ki = 25.12 nM T67162 CJ50AI 44212312 Ki = 199.53 nM T67162 CXR6K7 44212701 Ki > 1000 nM T67162 C8ORL9 44212702 Ki > 1000 nM T67162 CN71EI 44212703 Ki > 1000 nM T67162 CDO0I4 44214764 Ki = 8000 nM T67162 CK01JN 44214765 Ki = 5000 nM T67162 C9H3EV 44214766 Ki = 840 nM T67162 C7VWY4 44214767 Ki = 1200 nM T67162 CX54AP 44215433 Ki = 42 nM T67162 CT29ZS 44216196 Ki = 863 nM T67162 COS94W 44222483 Ki = 1.4 nM T67162 CNW3R8 44222488 Ki = 160 nM T67162 C1ST2I 44241718 Ki = 150 nM T67162 CJ8RW5 44249745 Ki = 42 nM T67162 C2FDB1 44250364 IC50 > 10000 nM T67162 C8MC0Q 44251387 IC50 > 10000 nM T67162 C5YEA8 44251388 IC50 > 10000 nM T67162 C0BSF6 44251389 IC50 > 10000 nM T67162 C2K0VZ 44253016 Ki > 1258.93 nM T67162 CT8MG3 44266611 Ki = 392 nM T67162 CFQ4L9 44266612 Ki = 93 nM T67162 C4QVN3 44266613 Ki = 77 nM T67162 C7AWM2 44266623 Ki = 50 nM T67162 CZ36NP 44266636 Ki = 4.1 nM T67162 CP52AC 44266663 Ki = 59 nM T67162 C5RH3X 44266664 Ki = 6.7 nM T67162 CIO03X 44266677 Ki = 108 nM T67162 CW14OJ 44266678 Ki > 339 nM T67162 CN90JC 44266689 Ki = 78 nM T67162 CFEI56 44267161 IC50 = 1778.28 nM T67162 CIZ5W7 44267181 IC50 = 2570.4 nM T67162 CGA1W5 44269820 Ki = 31 nM T67162 C0C4QN 44269825 Ki = 62 nM T67162 C43LUM 44270444 Ki = 12000 nM T67162 CWK09J 44270558 Ki = 4897.79 nM T67162 C1WZB8 44273552 Ki = 1584.89 nM T67162 CU8Y6L 44273553 Ki = 398.11 nM T67162 C28FOS 44273715 Ki = 1995.26 nM T67162 C2TN6O 44273720 Ki = 1000 nM T67162 CQV2Y7 44273741 Ki = 630.96 nM T67162 CUK3H6 44273815 Ki = 794.33 nM T67162 C7Z6BK 44273855 Ki = 158.49 nM T67162 CT9ZA7 44273876 Ki = 398.11 nM T67162 CFBT63 44273877 Ki = 1995.26 nM T67162 CPG2K5 44273882 Ki = 3981.07 nM T67162 C7H4GN 44273884 Ki = 251.19 nM T67162 C5DAM2 44273887 Ki = 2511.89 nM T67162 CDE2S1 44273896 Ki = 63.1 nM T67162 C2OMI3 44273897 Ki = 1584.89 nM T67162 C3J0GV 44273908 Ki = 794.33 nM T67162 CY2G0T 44273912 Ki = 1584.89 nM T67162 CG1L2J 44273920 Ki = 398.11 nM T67162 CMKG67 44273921 Ki = 1584.89 nM T67162 CX5PF6 44273924 Ki = 2511.89 nM T67162 CMW36L 44273925 Ki < 10000 nM T67162 CUP96S 44273927 Ki = 1584.89 nM T67162 CF46KT 44273928 Ki = 1000 nM T67162 CK7A9H 44274130 Ki = 79.43 nM T67162 CSIM26 44274174 Ki = 316.23 nM T67162 CQD08W 44274186 Ki = 3162.28 nM T67162 CQ83VT 44274687 Ki = 58 nM T67162 C4MHT3 44274739 Ki = 235 nM T67162 CLG10Y 44275015 Ki = 917 nM T67162 CSY7E4 44275135 Ki = 2.4 nM T67162 CVUE38 44275155 Ki = 100 nM T67162 C86EDH 44275362 Ki = 1.4 nM T67162 CBV7O8 44275604 Ki = 3.5 nM T67162 CE60XZ 44275616 Ki = 0.6 nM T67162 C1H0XC 44275766 Ki = 0.8 nM T67162 CMI4G9 44275820 Ki = 6512 nM T67162 CFP7Z8 44276050 Ki = 341 nM T67162 CE10KM 44276075 Ki = 726 nM T67162 CTM39J 44276079 Ki = 5148 nM T67162 CQ8V6N 44276105 Ki = 2108 nM T67162 C3AS0H 44276111 Ki = 95 nM T67162 C79YQZ 44276404 Ki = 1300 nM T67162 CWG0B7 44276405 Ki = 3600 nM T67162 CWS4K2 44276412 Ki = 1400 nM T67162 CNT6P3 44276414 Ki = 2200 nM T67162 CJEB02 44276535 Ki = 12000 nM T67162 CK2R3A 44276536 Ki = 168 nM T67162 CGC3Z5 44276551 Ki = 450 nM T67162 CHG9P5 44276552 Ki = 520 nM T67162 CT6XU0 44276556 Ki = 4400 nM T67162 C95QZD 44276557 Ki = 400 nM T67162 CTUC23 44276572 Ki = 890 nM T67162 CNHE76 44276598 Ki = 105 nM T67162 CLH93D 44276651 Ki = 9100 nM T67162 CTC47W 44276652 Ki = 1900 nM T67162 C0JPB1 44277402 Ki = 1288 nM T67162 CSB0G2 44277403 Ki = 151 nM T67162 CN1X3R 44277404 Ki = 5692 nM T67162 CX9PO7 44277421 Ki = 1288 nM T67162 CGD2I6 44277524 Ki = 996 nM T67162 CQV0T7 44277529 Ki = 2529 nM T67162 CXLV91 44277535 Ki = 1207 nM T67162 C27ULI 44277569 Ki > 10000 nM T67162 CF28KD 44277580 Ki = 7000 nM T67162 C4RG7F 44277587 Ki > 10000 nM T67162 C4HWK2 44277588 Ki > 10000 nM T67162 CGY34K 44277819 Ki = 5692 nM T67162 C84TMG 44278427 Ki = 709 nM T67162 CI37UT 44278788 Ki = 911 nM T67162 C3UK0D 44278789 Ki = 2336 nM T67162 CG0F7S 44282985 EC50 = 100 nM T67162 C8Q5RI 44283757 Ki = 1209 nM T67162 C1T2BY 44283889 Ki > 5000 nM T67162 CZF8B5 44283891 Ki > 5000 nM T67162 C5WHP1 44283941 Ki > 5000 nM T67162 CL3O5W 44286891 Ki = 47.5 nM T67162 C8J5HB 44286901 Ki = 763 nM T67162 C3YA5D 44286909 Ki > 1000 nM T67162 CAE7M3 44286910 Ki > 1000 nM T67162 CND65W 44287035 Ki = 1090 nM T67162 CON20Z 44287180 Ki > 1000 nM T67162 C17MSN 44287224 Ki = 1360 nM T67162 CARI13 44287238 Ki > 1000 nM T67162 CD9MT0 44287265 Ki > 1000 nM T67162 CRG2K4 44287274 Ki > 1000 nM T67162 C3TEZ8 44287301 Ki > 1000 nM T67162 CU50XS 44287333 Ki = 398 nM T67162 CE6C0P 44290360 Ki > 10000 nM T67162 CX87NU 44290508 Ki > 10000 nM T67162 CJI05D 44290522 Ki > 10000 nM T67162 CK5TX4 44297323 Ki = 251.19 nM T67162 C5NK9B 44297390 Ki = 1000 nM T67162 CSKN61 44297458 Ki = 501.19 nM T67162 CZR0L7 44297472 Ki = 316.23 nM T67162 C4G8QT 44297494 Ki = 316.23 nM T67162 CL5H8S 44297514 Ki = 158.49 nM T67162 CTK86W 44297596 Ki = 1584.89 nM T67162 CJD36K 44297665 Ki = 501.19 nM T67162 C5U0KI 44297693 Ki = 125.89 nM T67162 CWNI02 44297694 Ki = 100 nM T67162 C5X1PJ 44297720 Ki = 1000 nM T67162 CBSQ04 44300865 Ki = 170 nM T67162 CQ5A2E 44301054 Ki = 3700 nM T67162 CZ59OL 44301157 Ki = 1995.26 nM T67162 CNW2F3 44304314 IC50 = 2300 nM T67162 CWJA31 44304603 Ki = 280 nM T67162 CK8QJ6 44304621 Ki = 1070 nM T67162 CR9SB5 44304643 Ki = 3250 nM T67162 CH6FM8 44304644 Ki = 2750 nM T67162 CGY80N 44304652 Ki = 5050 nM T67162 CKBE16 44304814 Ki = 17500 nM T67162 C61YBG 44305039 Ki = 25.12 nM T67162 CIC7S0 44305123 Ki = 31.62 nM T67162 CHEO59 44305138 Ki = 501.19 nM T67162 C1V7ER 44305156 Ki = 25.12 nM T67162 C74GBN 44305165 Ki = 17 nM T67162 CJU47S 44305180 Ki = 423 nM T67162 C2XMP1 44305196 Ki = 10 nM T67162 CKX85J 44305348 Ki = 19.95 nM T67162 CU7J1E 44305390 Ki = 50.12 nM T67162 C2C8LF 44307285 Ki > 1000 nM T67162 C7EJ1R 44307286 Ki > 1000 nM T67162 CJ2QR0 44307437 Ki > 1000 nM T67162 CFBL97 44307498 Ki > 1000 nM T67162 CTI68M 44307546 Ki > 1000 nM T67162 CFDV86 44307552 Ki > 1000 nM T67162 CA3EG2 44307692 Ki > 1000 nM T67162 CQH1V4 44308839 Ki = 152 nM T67162 CMXV70 44308898 Ki = 6.35 nM T67162 CL3XD0 44309005 Ki = 22 nM T67162 CT2QB4 44309058 Ki = 118 nM T67162 CGYS61 44309076 Ki = 43.8 nM T67162 CB2HT7 44309448 Ki > 10000 nM T67162 CT1E5L 44309453 Ki = 10000 nM T67162 C9Y7AI 44309455 Ki = 47 nM T67162 C7HA6I 44309464 Ki > 10000 nM T67162 CJN2V0 44309466 Ki = 8400 nM T67162 C38TNP 44309468 Ki = 10000 nM T67162 C74QMW 44309492 Ki > 10000 nM T67162 CGP8X5 44309509 Ki = 29.6 nM T67162 CM92JC 44309510 Ki = 39.3 nM T67162 C70WAV 44309628 Ki = 10000 nM T67162 CP1QG5 44309688 Ki = 62.9 nM T67162 C1Q4JD 44309690 Ki > 10000 nM T67162 C1MH5F 44309692 Ki = 3130 nM T67162 CL3F0P 44309694 Ki = 2070 nM T67162 CA98DZ 44309696 Ki = 217 nM T67162 C0QFX9 44309716 Ki = 153 nM T67162 CKY68S 44309775 Ki = 168 nM T67162 C3YF2M 44309781 Ki = 2420 nM T67162 CX5DU2 44309807 Ki = 2110 nM T67162 CN0CZ1 44309809 Ki = 2600 nM T67162 CMJ95H 44309824 Ki > 10000 nM T67162 CV65SY 44309831 Ki = 70 nM T67162 CX8H4A 44309835 Ki = 152 nM T67162 CT8L0X 44309837 Ki = 20000 nM T67162 CG97RP 44309852 Ki > 10000 nM T67162 CT37BP 44309854 Ki > 10000 nM T67162 CE2QW0 44309866 Ki > 10000 nM T67162 C1TKV6 44309876 Ki = 36.8 nM T67162 C51RVN 44309974 Ki = 2690 nM T67162 CCQN61 44309978 Ki = 5320 nM T67162 C4UZG0 44309993 Ki = 7180 nM T67162 CLYS40 44309995 Ki > 10000 nM T67162 CH86ST 44310013 Ki = 2900 nM T67162 C9LHD4 44310018 Ki = 10000 nM T67162 CUC5I7 44310027 Ki = 550 nM T67162 C03FIO 44310034 Ki > 10000 nM T67162 CU0EA9 44310036 Ki > 10000 nM T67162 CJYR45 44310038 Ki = 10000 nM T67162 C7M5HP 44310050 Ki = 1656 nM T67162 C09JTN 44310052 Ki = 1420 nM T67162 C4MD0R 44310071 Ki = 962 nM T67162 CY6O4H 44310073 Ki = 642 nM T67162 CN19YU 44310110 Ki = 32000 nM T67162 CL8D2O 44310124 Ki = 7630 nM T67162 C4FS9Q 44310126 Ki = 4870 nM T67162 CKVO42 44310128 Ki = 24000 nM T67162 CI2TN6 44310145 Ki = 2370 nM T67162 CRD9Z2 44310792 Ki = 398.11 nM T67162 C9GLP3 44311009 Ki = 100 nM T67162 C42QYO 44311177 Ki > 100000 nM T67162 C6BX5O 44311179 Ki = 1496 nM T67162 C6HEB9 44311180 Ki > 10000 nM T67162 C02DAJ 44311195 Ki = 1460 nM T67162 CH7Q9A 44311197 Ki = 2030 nM T67162 CBZ06X 44311211 Ki = 2330 nM T67162 C5YNX7 44311359 Ki > 10000 nM T67162 C6D5TP 44311361 Ki > 10000 nM T67162 C7VW2Z 44311445 Ki > 100000 nM T67162 C71HBP 44311480 Ki = 2900 nM T67162 CRW2P1 44311482 Ki = 1080 nM T67162 CCNT08 44311493 Ki = 4100 nM T67162 CW8S4Z 44311613 Ki = 1530 nM T67162 CO2P4D 44311615 Ki = 7600 nM T67162 C3QI6S 44311621 Ki = 4200 nM T67162 CTR73J 44311625 Ki > 10000 nM T67162 C5IKM9 44311640 Ki = 8780 nM T67162 C8JP5T 44315098 Ki = 3 nM T67162 CN9ZV0 44315099 Ki = 1.3 nM T67162 C9BTW3 44315120 Ki = 10 nM T67162 CFB13Y 44315131 Ki = 12 nM T67162 CJL61P 44315181 Ki > 10000 nM T67162 CYVZ78 44315380 Ki = 2.2 nM T67162 C6AWP3 44315381 Ki = 0.93 nM T67162 C83WGQ 44315382 Ki = 1 nM T67162 CP9D6G 44315383 Ki = 4 nM T67162 CV4X1P 44315386 Ki = 10 nM T67162 CU4V7O 44315403 Ki > 10000 nM T67162 C9G2KL 44315406 Ki = 0.41 nM T67162 C2HUA3 44315407 Ki = 10 nM T67162 CHJ1I7 44315426 Ki = 18 nM T67162 CFE15Q 44315427 Ki = 8.1 nM T67162 C8S5RH 44315436 Ki = 2 nM T67162 CL0Z3J 44315453 Ki = 6 nM T67162 CLCN19 44315510 Ki > 10000 nM T67162 CC57FY 44315535 Ki > 10000 nM T67162 CEU56A 44315536 Ki > 10000 nM T67162 C2DB7M 44315537 Ki = 1837 nM T67162 CF3VK8 44315548 Ki = 4.6 nM T67162 C06BLA 44315552 Ki = 1356 nM T67162 C49OQD 44315568 Ki = 8.1 nM T67162 C7TCE9 44315569 Ki = 9.3 nM T67162 CI9GC2 44315578 Ki > 10000 nM T67162 CW2I9R 44315579 Ki = 4324 nM T67162 CF3M9C 44315580 Ki = 2183 nM T67162 CSF86X 44315581 Ki = 1062 nM T67162 CJ78AN 44315794 Ki > 10000 nM T67162 C6B4CM 44315795 Ki = 620 nM T67162 C2WNL8 44315815 Ki > 10000 nM T67162 CMRY42 44315830 Ki = 948 nM T67162 C6RF1P 44316315 Ki = 130 nM T67162 CL6KC8 44317000 Ki = 339 nM T67162 CRIT59 44317001 Ki = 10 nM T67162 C47HKR 44317002 Ki = 19 nM T67162 C60LKZ 44317003 Ki = 11.4 nM T67162 CL3B1F 44317030 Ki = 16.5 nM T67162 C2J1GU 44317031 Ki = 6.3 nM T67162 C9LF3J 44317054 Ki = 6.5 nM T67162 C2XY0L 44317069 Ki = 5 nM T67162 C1HK5Z 44317088 Ki = 34 nM T67162 C1VLM3 44317105 Ki = 1 nM T67162 CG9FT0 44317222 Ki = 182 nM T67162 C6JMU9 44317229 Ki = 16.5 nM T67162 CA2ZM7 44317252 Ki = 37.5 nM T67162 CXK60V 44317260 Ki = 81 nM T67162 C3CZD1 44317272 Ki = 4.5 nM T67162 C9ZK2O 44317275 Ki = 15 nM T67162 C6TC3I 44317294 Ki = 5 nM T67162 C9DKH3 44317295 Ki = 5.6 nM T67162 CVP35Q 44317384 Ki = 12 nM T67162 CO6I2J 44317385 Ki = 1.4 nM T67162 CZ6O2I 44317425 Ki = 10 nM T67162 CDI5G8 44317436 Ki = 12 nM T67162 CT7S5Y 44317450 Ki = 1.7 nM T67162 CBW78P 44317467 Ki = 3 nM T67162 CTFO42 44317468 Ki = 177 nM T67162 CV8WZ0 44318454 IC50 = 36.31 nM T67162 CXJL56 44318842 IC50 = 54.95 nM T67162 CWUE26 44319102 Ki = 330 nM T67162 CTE14R 44319217 Ki = 126 nM T67162 C8LXY4 44319269 Ki = 1518 nM T67162 CV2UN7 44319361 Ki = 720 nM T67162 CN1M5O 44319362 Ki > 3333 nM T67162 CC2W9S 44319368 Ki = 110 nM T67162 CCD3V1 44319369 Ki = 320 nM T67162 CY9ZX7 44319370 Ki = 2400 nM T67162 CUB9J4 44319412 Ki > 3333 nM T67162 C3Z9BT 44319418 Ki = 3945 nM T67162 C82GVM 44319482 Ki > 3333 nM T67162 CC2GZ0 44319568 Ki = 803 nM T67162 C31IGQ 44319569 Ki = 1750 nM T67162 CJ02KH 44319612 Ki = 1027 nM T67162 CK0D6E 44319723 Ki = 199.53 nM T67162 CU06KP 44319980 Ki = 316.23 nM T67162 CHT83A 44320347 Ki = 11 nM T67162 CG5E2U 44323763 Ki = 4.1 nM T67162 CY1I0M 44323780 Ki = 540 nM T67162 C5CP2K 44323851 Ki = 57 nM T67162 CVZ27T 44323870 Ki = 690 nM T67162 CNYT01 44323874 Ki = 150 nM T67162 CHE75M 44323876 Ki = 290 nM T67162 CAO54X 44323890 Ki = 730 nM T67162 C7Y5PV 44323894 Ki = 94 nM T67162 C4KGL6 44324017 Ki = 85 nM T67162 C2MSG8 44324041 Ki = 39 nM T67162 CY03UK 44324042 Ki = 68 nM T67162 C5IFM9 44324046 Ki = 17 nM T67162 CE3BO7 44324047 Ki = 0.42 nM T67162 C3C5LO 44324051 Ki = 187 nM T67162 C1NFW3 44324052 Ki = 17 nM T67162 C2W0VB 44324056 Ki = 250 nM T67162 CT48CS 44324065 Ki = 92 nM T67162 C9UR6K 44324070 Ki = 78 nM T67162 CO25PJ 44324071 Ki > 1000 nM T67162 CPZ7N8 44324079 Ki = 290 nM T67162 CF72QK 44324084 Ki = 3000 nM T67162 CM45XW 44324091 Ki = 21 nM T67162 CW16JD 44324737 Ki > 1000 nM T67162 CA84SN 44324765 Ki = 959 nM T67162 COA3H4 44324800 Ki = 230 nM T67162 CLDK96 44324801 Ki = 1258.93 nM T67162 C2SMT6 44324802 Ki = 1584.89 nM T67162 CY04JW 44324972 Ki > 1000 nM T67162 C3UWI1 44324978 Ki = 1584.89 nM T67162 C0Z1NV 44324979 Ki = 2511.89 nM T67162 CCT67J 44324980 Ki = 42 nM T67162 CB5H2S 44324986 Ki = 501.19 nM T67162 CUZ67X 44325021 Ki = 1584.89 nM T67162 CN07UQ 44325025 Ki = 158.49 nM T67162 CI30DU 44325026 Ki = 2511.89 nM T67162 C8KWG4 44325037 Ki = 1258.93 nM T67162 CGL51N 44325577 Ki > 217 nM T67162 CXPS18 44325578 Ki > 217 nM T67162 COM07T 44325658 Ki > 217 nM T67162 CQE81D 44325894 Ki > 217 nM T67162 CE0S1Z 44325900 Ki > 217 nM T67162 CKW98Z 44325908 Ki = 11 nM T67162 C5VLY2 44326733 Ki = 4600 nM T67162 C1Y4VO 44329046 Ki = 1995.26 nM T67162 C69IHO 44329050 Ki = 794.33 nM T67162 CFA61T 44329053 Ki = 630.96 nM T67162 CZX74M 44329058 Ki = 398.11 nM T67162 CT8KH0 44329062 Ki = 794.33 nM T67162 C5NOQ0 44329068 Ki = 501.19 nM T67162 CM9NS0 44329102 Ki = 501.19 nM T67162 CI2Z9F 44329106 Ki = 251.19 nM T67162 COL9X4 44329121 Ki = 1258.93 nM T67162 C5QOA8 44329126 Ki = 1000 nM T67162 CT7CZ6 44329130 Ki = 316.23 nM T67162 CR5FP1 44329136 Ki = 630.96 nM T67162 C1WYS3 44329321 Ki = 25 nM T67162 C90PLN 44329483 Ki = 197 nM T67162 C5J3PW 44329749 Ki = 533 nM T67162 C6NH5U 44329754 Ki > 10000 nM T67162 C5U1WN 44330292 Ki > 10000 nM T67162 C4P1XE 44330386 Ki = 534 nM T67162 CIWY10 44330417 Ki > 10000 nM T67162 CROD75 44330514 Ki = 555 nM T67162 C1UTG6 44330515 Ki > 10000 nM T67162 CFI52O 44330553 Ki = 28 nM T67162 C12EKB 44330564 Ki > 10000 nM T67162 COK95B 44330566 Ki = 489 nM T67162 C3DOY1 44330567 Ki = 416 nM T67162 CQRP49 44330574 Ki > 10000 nM T67162 CZPL05 44330585 Ki > 10000 nM T67162 C0RX1F 44330637 Ki > 10000 nM T67162 C7CNK8 44330638 Ki > 10000 nM T67162 C4JP8S 44330639 Ki > 10000 nM T67162 CJZQ05 44330640 Ki > 10000 nM T67162 C98JGO 44330650 Ki > 10000 nM T67162 C26UAW 44330694 Ki = 885 nM T67162 CYP6M3 44331310 Ki = 510 nM T67162 C6H4BO 44332565 Ki = 75.8 nM T67162 C9JQK3 44332566 Ki > 1000 nM T67162 C1E7KI 44332581 Ki = 456 nM T67162 CD7N6W 44332613 Ki > 300 nM T67162 COR0D5 44332646 Ki > 10000 nM T67162 C63TDB 44332686 Ki = 37.6 nM T67162 COG5D1 44332701 Ki = 9 nM T67162 CZ6F4T 44333001 Ki = 375 nM T67162 C0UT6E 44333374 Ki = 630 nM T67162 C9MVH8 44333746 Ki > 4780 nM T67162 C2YZI8 44334603 Ki = 6.7 nM T67162 C1DH4T 44334637 Ki = 0.2 nM T67162 CK1UB8 44335678 Ki = 1414 nM T67162 CRD80K 44335721 Ki = 2552 nM T67162 CIMQ72 44335722 Ki = 3431 nM T67162 CO6YN8 44335739 Ki = 23 nM T67162 CRL68J 44335746 Ki = 3011 nM T67162 C7AN0J 44335761 Ki = 225 nM T67162 CS4A3Z 44335795 Ki = 166 nM T67162 CL1BV7 44335796 Ki = 62 nM T67162 CJ98HN 44335798 Ki = 1530 nM T67162 CT54MD 44335799 Ki = 620 nM T67162 C7FYS0 44335800 Ki = 2094 nM T67162 C3I6KY 44335812 Ki = 39 nM T67162 C3YNI6 44335813 Ki = 834 nM T67162 C7Y2LT 44335816 Ki = 3823 nM T67162 CB15TR 44335828 Ki = 1918 nM T67162 CNZ0F5 44335829 Ki = 1784 nM T67162 COS7V9 44335835 Ki = 5940 nM T67162 CYIF05 44335847 Ki = 2364 nM T67162 CM85JR 44335853 Ki = 5287 nM T67162 C0A5DO 44335876 Ki = 119 nM T67162 CYE80K 44335877 Ki = 2583 nM T67162 CLW0Z6 44335884 Ki = 71 nM T67162 C6WA4H 44335886 Ki = 52 nM T67162 CX8AZ4 44335889 Ki = 713 nM T67162 CCJ38R 44335893 Ki = 199 nM T67162 C0XR3S 44335896 Ki = 1692 nM T67162 CQ2U5E 44335907 Ki = 214 nM T67162 C2D5HQ 44335908 Ki = 218 nM T67162 CR31UG 44335909 Ki = 134 nM T67162 C08FAK 44335918 Ki = 491 nM T67162 C85UNM 44335919 Ki = 96 nM T67162 CG6K4D 44335923 Ki = 753 nM T67162 C3EIN8 44335924 Ki = 887 nM T67162 C2A3OP 44335925 Ki = 28 nM T67162 CA2UE5 44335945 Ki > 1000 nM T67162 C6YM5Z 44335960 Ki = 191 nM T67162 CA1T9Z 44335971 Ki = 1252 nM T67162 CT78OA 44335972 Ki = 5247 nM T67162 C75EDP 44335973 Ki = 95 nM T67162 C5ZRM3 44335979 Ki = 6357 nM T67162 C69XES 44335987 Ki = 35 nM T67162 CEV25H 44335991 Ki > 10000 nM T67162 CSWA61 44335995 Ki = 219 nM T67162 CUK23N 44335996 Ki = 43 nM T67162 CZD10E 44335998 Ki > 1000 nM T67162 CK1I5J 44336000 Ki = 1149 nM T67162 C0AY1E 44336003 Ki = 5847 nM T67162 COK93P 44336004 Ki = 1926 nM T67162 C0QH8A 44336005 Ki = 2220 nM T67162 C3QW4H 44336006 Ki = 1207 nM T67162 CX2L3Z 44336012 Ki = 747 nM T67162 CR4B0K 44336018 Ki > 1000 nM T67162 CR4SU0 44336027 Ki = 1000 nM T67162 CG8U9R 44336030 Ki = 758 nM T67162 CHE0R6 44336035 Ki = 2145 nM T67162 CQ38GM 44336036 Ki = 5839 nM T67162 C3KV9L 44336045 Ki = 8620 nM T67162 C3EF1C 44336046 Ki = 4742 nM T67162 C5H1SL 44336047 Ki = 286 nM T67162 CRIF94 44336050 Ki = 306 nM T67162 CY60UT 44336051 Ki = 120 nM T67162 CL0HI9 44336052 Ki = 6740 nM T67162 CO4M5K 44336055 Ki = 4126 nM T67162 CJLR98 44336057 Ki = 3325 nM T67162 C4W8NC 44336059 Ki > 1000 nM T67162 C7OW8Y 44336061 Ki = 113 nM T67162 CYP35N 44336062 Ki = 9395 nM T67162 CK1IQ0 44336074 Ki > 10000 nM T67162 C6K9QY 44336075 Ki = 158 nM T67162 CD80AW 44336085 Ki > 5000 nM T67162 CN4A2F 44336099 Ki = 271 nM T67162 CUQS13 44336100 Ki = 377 nM T67162 CP3HA8 44336105 Ki = 341 nM T67162 CK4H8R 44336108 Ki = 509 nM T67162 CDY2E4 44336109 Ki = 518 nM T67162 CFZ9U0 44336127 Ki = 2524 nM T67162 CIB45H 44336138 Ki = 979 nM T67162 CJR1X5 44336154 Ki = 883 nM T67162 CX8EA2 44336172 Ki = 3780 nM T67162 CJ4F0T 44336175 Ki = 487 nM T67162 CJB61S 44336194 Ki = 3780 nM T67162 CS7G8O 44336313 Ki > 1000 nM T67162 C1YIQ4 44336314 Ki = 1642 nM T67162 C26ZUF 44336352 Ki = 129 nM T67162 CFT4L1 44336552 Ki = 7800 nM T67162 CS3TZ4 44336571 Ki = 13000 nM T67162 CT3M2R 44337675 Ki = 180 nM T67162 C2ECI8 44337709 Ki = 1120 nM T67162 C5S9WU 44337725 Ki = 672 nM T67162 C9ZH7J 44338130 Ki = 2600 nM T67162 C0ZH4Y 44338149 Ki = 927 nM T67162 CH2VD3 44338186 Ki = 550 nM T67162 CXPZ62 44338224 Ki = 1200 nM T67162 CPW0H6 44338236 Ki = 1100 nM T67162 CXEQ14 44338237 Ki = 800 nM T67162 CQ0ZF9 44338248 Ki = 218 nM T67162 C92LYP 44338257 Ki = 4200 nM T67162 C7CKX5 44338263 Ki = 270 nM T67162 CQHD85 44338264 Ki = 310 nM T67162 CW8A4D 44338272 Ki = 330 nM T67162 CYP6X3 44338285 Ki = 300 nM T67162 C8R3HT 44338286 Ki = 140 nM T67162 CX5Y0E 44338291 Ki = 550 nM T67162 CW0EV9 44338292 Ki = 800 nM T67162 CWM3S8 44338297 Ki = 6200 nM T67162 CGET31 44338308 Ki = 1500 nM T67162 CVZM05 44338310 Ki = 38 nM T67162 C85MCE 44338319 Ki = 1100 nM T67162 CC1D4E 44338326 Ki = 24 nM T67162 CV37EY 44338387 Ki = 73 nM T67162 C2ODN5 44338389 Ki = 1100 nM T67162 CWYD83 44338402 Ki > 43000 nM T67162 CWKN28 44339794 IC50 > 1000 nM T67162 C1I8XF 44339879 Ki = 130 nM T67162 C34CBZ 44339953 Ki = 7.4 nM T67162 CPF62D 44339984 Ki = 260 nM T67162 CIS79K 44339992 Ki = 135 nM T67162 C84OZX 44340084 Ki = 6.4 nM T67162 C9I7GN 44340097 Ki = 11 nM T67162 CBQ3D5 44340186 Ki = 1100 nM T67162 CT5HC3 44340227 Ki = 23 nM T67162 C7-SEP 44340278 Ki = 39.81 nM T67162 C1EZY8 44340285 Ki = 6.31 nM T67162 C6LDF1 44340301 Ki = 100 nM T67162 C5HGU2 44340302 Ki = 1900 nM T67162 CA71HQ 44340333 Ki = 82 nM T67162 CJL8H0 44340337 Ki = 15.85 nM T67162 C8RN4J 44340352 Ki = 7.943 nM T67162 CFRK78 44340353 Ki = 39.81 nM T67162 CUG2V9 44340354 Ki = 25.12 nM T67162 CA1F3K 44340364 Ki = 19.95 nM T67162 CQPW26 44340376 Ki = 420 nM T67162 C3QW1F 44340415 Ki = 4000 nM T67162 CO2QV3 44340654 Ki = 25.12 nM T67162 CLK24X 44340661 Ki = 794.33 nM T67162 C8FC4J 44340690 Ki = 10 nM T67162 C2N0UR 44340694 Ki = 1258.93 nM T67162 CPOL72 44340695 Ki = 3.162 nM T67162 CS48JN 44340705 Ki = 31.62 nM T67162 C26ITO 44340881 IC50 > 10000 nM T67162 CF94RB 44340893 IC50 > 10000 nM T67162 C6HED7 44340900 IC50 = 4100 nM T67162 CQ2M3C 44340915 IC50 = 1500 nM T67162 CXKI34 44340919 IC50 = 4900 nM T67162 CUW0O9 44340942 IC50 = 2500 nM T67162 CWZ0D7 44340945 IC50 = 890 nM T67162 C8QYA4 44340965 Ki = 0.3981 nM T67162 CC2D6N 44340967 Ki = 1 nM T67162 CB2G0T 44340985 Ki = 79.43 nM T67162 CP9J2Y 44341034 IC50 > 10000 nM T67162 C1L8EB 44341173 IC50 > 10000 nM T67162 CK46JF 44341181 IC50 = 7100 nM T67162 CD9ZS8 44342270 IC50 = 480 nM T67162 CH69UL 44344506 Ki > 1000 nM T67162 C6N3XK 44345317 IC50 < 1000 nM T67162 C8R4YG 44347445 Ki = 541 nM T67162 CZV21Q 44347713 Ki = 776 nM T67162 CLG65Q 44347771 Ki = 202 nM T67162 CUI12W 44347787 Ki > 10000 nM T67162 C7Q4IB 44347788 Ki > 10000 nM T67162 CCU89V 44350664 Ki = 124.4 nM T67162 C5GW8X 44350679 Ki = 50 nM T67162 CTXY90 44350788 Ki = 19.5 nM T67162 CZX4S1 44350839 Ki = 53.2 nM T67162 C4QP5U 44350942 Ki = 101 nM T67162 C50HVX 44350991 Ki = 403 nM T67162 CUGT13 44351005 EC50 = 2.5 nM T67162 C02OXY 44353233 Ki = 20 nM T67162 CNVZ48 44353234 Ki = 20 nM T67162 CEW8G9 44353236 Ki = 25 nM T67162 CNC65I 44353323 Ki = 40 nM T67162 C8SX6R 44353325 Ki = 125.89 nM T67162 CKEG16 44353327 Ki = 25 nM T67162 CR2F9X 44353343 Ki = 40 nM T67162 C0ZYJ5 44353345 Ki = 398.11 nM T67162 CFIO91 44353352 Ki = 316.23 nM T67162 C65MOI 44353353 Ki = 794.33 nM T67162 C06VLC 44353354 Ki = 125.89 nM T67162 CAF53W 44353361 Ki = 6309.57 nM T67162 CI2HW1 44353363 Ki = 1000 nM T67162 CH94PY 44353393 Ki = 630.96 nM T67162 CGA62E 44353398 Ki = 316.23 nM T67162 CX02GJ 44353399 Ki = 630.96 nM T67162 CVK1R7 44353406 Ki = 794.33 nM T67162 CR7V1I 44353412 Ki = 251.19 nM T67162 C3CA9O 44353413 Ki = 25 nM T67162 CT6HG1 44353414 Ki = 25 nM T67162 CM1Y8U 44353431 Ki = 316.23 nM T67162 CAQC14 44353432 Ki = 100 nM T67162 CULV76 44353438 Ki = 1000 nM T67162 CI3QT4 44353445 Ki = 10 nM T67162 COQ4U3 44353459 Ki = 12 nM T67162 CPU2L5 44353461 Ki = 40 nM T67162 C4WIZ8 44353462 Ki = 100 nM T67162 CWX5J3 44353475 Ki = 251.19 nM T67162 CJ0AS5 44353476 Ki = 398.11 nM T67162 CEOI46 44353477 Ki = 794.33 nM T67162 CDK4M0 44353487 Ki = 199.53 nM T67162 CU67QT 44353488 Ki = 199.53 nM T67162 CNF6G0 44353492 Ki = 40 nM T67162 CZV3S0 44355355 Ki = 250 nM T67162 CNV5M9 44355433 Ki = 1046 nM T67162 C9W5AB 44356064 Ki = 550 nM T67162 C9GB5E 44356253 Ki = 4.3 nM T67162 CKL64H 44358192 Ki = 2 nM T67162 CJ80OW 44360984 Ki = 180 nM T67162 CS8K1A 44360992 Ki = 34 nM T67162 C3NZ7B 44361021 Ki = 58 nM T67162 CL2RI0 44363213 Ki = 199.53 nM T67162 C8WJ7M 44363215 Ki = 501.19 nM T67162 CIS8Z4 44363218 Ki = 398.11 nM T67162 COY57L 44363232 Ki = 1000 nM T67162 CTM6J0 44363348 Ki = 125.89 nM T67162 CPO24U 44363755 IC50 = 761 nM T67162 CMU02Q 44364616 Ki = 570 nM T67162 C9WC1P 44365113 IC50 > 1000 nM T67162 CDQ75B 44365114 IC50 > 1000 nM T67162 C8LB3Y 44365166 Ki = 460 nM T67162 C7B6EY 44365175 Ki = 6.7 nM T67162 C4ZM9C 44365177 Ki = 120 nM T67162 C2WY0V 44365298 IC50 > 1000 nM T67162 CDC2Q4 44365299 IC50 > 1000 nM T67162 C5JLD7 44369020 Ki > 1000 nM T67162 CJ0SZ2 44369910 Ki = 194.98 nM T67162 CZIP61 44369921 Ki < 10000 nM T67162 CW2X3H 44369922 Ki = 398.11 nM T67162 CG5A2S 44369987 Ki = 107.15 nM T67162 CXIM47 44369992 Ki = 275.42 nM T67162 C9ZB4M 44370009 Ki = 600 nM T67162 C81CTM 44370032 Ki = 1300 nM T67162 C50OBQ 44370047 Ki = 800 nM T67162 C4JCY7 44370058 Ki = 900 nM T67162 C1U9IX 44370125 Ki < 10000 nM T67162 CM3W6Y 44370126 Ki = 223.87 nM T67162 C2SD5H 44370139 Ki = 831.76 nM T67162 C0DQS7 44371025 Ki = 622 nM T67162 CU49IQ 44371356 Ki = 354 nM T67162 CR5IM4 44371566 Ki = 782 nM T67162 C6PSR0 44371932 Ki = 9200 nM T67162 CQ1IU6 44371980 Ki = 120 nM T67162 C2JFZ9 44371996 Ki = 400 nM T67162 CK6GM7 44371997 Ki = 21000 nM T67162 CXZ6A7 44372009 Ki = 2800 nM T67162 C4VLE2 44372153 Ki = 24000 nM T67162 CJXL12 44372154 Ki = 14000 nM T67162 C4O3LX 44372198 Ki = 15000 nM T67162 C3QBW5 44372199 Ki = 0.031 nM T67162 CZV9O7 44372296 Ki = 22000 nM T67162 C1SWI7 44372312 Ki = 56000 nM T67162 CX2B6A 44372338 Ki = 2800 nM T67162 C3GJM6 44374188 Ki = 2511.89 nM T67162 CVL3U2 44374207 Ki > 1000 nM T67162 CV8CP3 44374225 Ki > 1000 nM T67162 C04WKH 44374233 Ki = 870 nM T67162 CJ4A2U 44374299 Ki > 1000 nM T67162 C39OSY 44374408 Ki = 2511.89 nM T67162 C6L9AR 44374409 Ki = 398.11 nM T67162 C20MKC 44374410 Ki = 199.53 nM T67162 CAJ92G 44374411 Ki = 100 nM T67162 CD5E1G 44374431 Ki = 2328 nM T67162 CK28HY 44374637 Ki = 546 nM T67162 C8EK9X 44374648 Ki = 2557 nM T67162 C4BAI3 44374753 IC50 > 10000 nM T67162 CPL87U 44374827 Ki = 26 nM T67162 CEC54D 44374863 Ki = 165 nM T67162 CNF12S 44376209 Ki = 68 nM T67162 CG1H4I 44376230 Ki = 1720 nM T67162 CGX1Z3 44376241 Ki = 918 nM T67162 C2UD1H 44376569 Ki = 38 nM T67162 CM57EJ 44376876 Ki = 44 nM T67162 C2S0TL 44376918 Ki = 187 nM T67162 CD2R5X 44376920 Ki = 948 nM T67162 CGX72S 44376921 Ki = 254 nM T67162 CVW0F4 44377901 Ki = 18 nM T67162 C2NE7B 44377927 Ki = 4 nM T67162 C1IDK8 44377928 Ki = 41 nM T67162 CD0T3J 44377939 Ki = 7.7 nM T67162 CN3FA5 44377954 Ki = 3.4 nM T67162 C49FLN 44377965 Ki = 15.1 nM T67162 CZK50H 44378001 Ki = 29 nM T67162 CVH02T 44378002 Ki = 63 nM T67162 C03SDF 44378003 Ki = 5.2 nM T67162 C62RSW 44378016 Ki = 68 nM T67162 C6Z9UH 44378022 Ki = 60 nM T67162 C7JB3Y 44378024 Ki = 23 nM T67162 C1UY7T 44378034 Ki = 14 nM T67162 C56ZJP 44378035 Ki = 19 nM T67162 CTC75H 44378076 Ki = 5.9 nM T67162 C3GTV5 44378077 Ki = 2.7 nM T67162 CS07QF 44378128 Ki = 17 nM T67162 CWU41H 44378141 Ki = 26 nM T67162 C9R5AX 44378333 Ki = 19 nM T67162 C6EMI4 44378348 Ki = 20 nM T67162 CJF5K0 44378369 Ki = 3.5 nM T67162 CJ3ZM8 44378381 Ki = 11 nM T67162 CYI39O 44380685 Ki = 540 nM T67162 CL1ER5 44380697 Ki = 640 nM T67162 C6B9PA 44380715 Ki = 58 nM T67162 CNSG64 44380716 Ki = 28000 nM T67162 C6MWD2 44380717 Ki = 19000 nM T67162 CA5EW9 44380770 Ki = 190 nM T67162 C68MUE 44380774 Ki = 10 nM T67162 C4DGR5 44380785 Ki = 21 nM T67162 CUV90Q 44380802 Ki = 120 nM T67162 CCL54M 44380815 Ki = 79 nM T67162 CM01SN 44380816 Ki = 1600 nM T67162 CT02DY 44380921 Ki = 540 nM T67162 C6PI1L 44381117 Ki = 25000 nM T67162 CJ6I0B 44381118 Ki = 86 nM T67162 CBYQ74 44381146 Ki = 19000 nM T67162 C8GA2E 44381147 Ki = 24 nM T67162 C6SDO5 44381216 Ki = 25000 nM T67162 C4OAD2 44381217 Ki = 43000 nM T67162 C67SRD 44381276 Ki = 6400 nM T67162 CKR9B8 44381279 Ki = 2800 nM T67162 COB6T7 44381286 Ki = 14000 nM T67162 CZ7Q2X 44381424 Ki = 4200 nM T67162 CQO5G1 44381432 Ki = 14000 nM T67162 CI0YA1 44382105 Ki < 100000 nM T67162 CPDA94 44382118 Ki = 5011.87 nM T67162 CRK0U1 44382163 Ki = 1000 nM T67162 CF7E9O 44382164 Ki = 398.11 nM T67162 C5CG2L 44382165 Ki = 2511.89 nM T67162 CSC5Z4 44382774 Ki < 10000 nM T67162 C7KW3P 44382826 Ki < 10000 nM T67162 CUL1Y2 44382827 Ki < 10000 nM T67162 C5H4KM 44382828 Ki = 501.19 nM T67162 C8L5WN 44382829 Ki = 12589.25 nM T67162 C1XOB5 44387732 Ki = 791 nM T67162 CL54KN 44387733 Ki = 266 nM T67162 C80WKC 44387740 Ki > 1500 nM T67162 CROA61 44387743 Ki = 2000 nM T67162 C1M5OY 44387746 Ki > 1000 nM T67162 CK36VZ 44387776 Ki > 2000 nM T67162 CC0WK5 44387777 Ki > 2000 nM T67162 CQ9WS8 44387780 Ki > 1000 nM T67162 CQ85AW 44389003 Ki > 2000 nM T67162 C8AG7U 44389016 Ki > 2000 nM T67162 CB8L9M 44389309 Ki = 21.2 nM T67162 CI5P0E 44389321 Ki = 6.2 nM T67162 CVYR53 44389330 Ki = 11.9 nM T67162 C1B0VT 44389345 Ki = 3.6 nM T67162 CT8Y5A 44393007 Ki > 1000 nM T67162 CE03ZW 44393134 Ki > 1000 nM T67162 CG5UE1 44393169 Ki > 1000 nM T67162 C6WAK2 44393173 Ki = 28.18 nM T67162 CK85EB 44393193 Ki > 1000 nM T67162 CEO2W9 44393372 Ki = 1 nM T67162 CXP4Q7 44393393 Ki = 32 nM T67162 C6BZS0 44393403 Ki = 27 nM T67162 C86NED 44393411 Ki = 140 nM T67162 C9THO4 44393415 Ki = 35 nM T67162 CQAS90 44394590 Ki = 900 nM T67162 CTB7O0 44394599 Ki = 3100 nM T67162 C4V1DZ 44394618 Ki = 120 nM T67162 C67SCU 44394629 Ki = 4000 nM T67162 CGC24Z 44394636 Ki = 1500 nM T67162 CSK9Z7 44394666 Ki = 1000 nM T67162 CL8C1E 44394667 Ki = 94 nM T67162 CW0M6Y 44394675 Ki = 3700 nM T67162 C1MC6J 44394742 Ki = 70 nM T67162 COD15M 44394743 Ki = 60 nM T67162 CBZU60 44394820 Ki = 4000 nM T67162 COU0F6 44394884 Ki = 150 nM T67162 C8EC7R 44395709 Ki = 1231 nM T67162 CF7I1C 44395711 Ki = 1050 nM T67162 C2KFE4 44395714 Ki = 189.8 nM T67162 C3RV6T 44395741 Ki = 29.51 nM T67162 C4B0OI 44397588 Ki = 794.33 nM T67162 C5FP0R 44397589 Ki = 1258.93 nM T67162 CE3G8U 44397670 Ki = 1258.93 nM T67162 C0E5HY 44400500 Ki = 45 nM T67162 CO8EU5 44400519 Ki = 12 nM T67162 CRX12E 44400553 Ki = 72 nM T67162 CIU18E 44400585 Ki = 60 nM T67162 CV8K2W 44400594 Ki = 120 nM T67162 C84RNU 44400626 Ki = 19 nM T67162 CY94SF 44400674 Ki = 78 nM T67162 CX7O9S 44401041 Ki = 32 nM T67162 C5XC2B 44401042 Ki = 68 nM T67162 CD56EA 44401105 Ki = 66 nM T67162 CW3PC2 44401106 Ki = 12 nM T67162 C9WH7P 44401164 Ki = 1.7 nM T67162 C9CWX1 44401194 Ki = 191 nM T67162 CXT84G 44401243 Ki = 5.9 nM T67162 CR7H0V 44401244 Ki = 369 nM T67162 C1B4QL 44403095 Ki > 10000 nM T67162 C1YL7Z 44403098 Ki > 10000 nM T67162 CFV98A 44403101 Ki > 10000 nM T67162 C6OY9S 44403102 Ki > 10000 nM T67162 CH4SX6 44403105 Ki > 10000 nM T67162 C12FIH 44403106 Ki > 10000 nM T67162 CQ4U2P 44403210 Ki = 98 nM T67162 CKE6T4 44403213 Ki = 17 nM T67162 CAJX39 44403214 Ki = 160 nM T67162 C61CNS 44403219 Ki = 21 nM T67162 C5AE9L 44403220 Ki = 260 nM T67162 CC6XM4 44403224 Ki = 44 nM T67162 C6JB4M 44403225 Ki = 72 nM T67162 CGE52H 44403232 Ki = 39 nM T67162 C4LKC1 44404394 Ki > 10000 nM T67162 C3EJ4G 44404396 Ki > 10000 nM T67162 C0E9YL 44404412 Ki = 25 nM T67162 CR3Q7O 44404413 Ki = 18 nM T67162 CGCW03 44404417 Ki = 17 nM T67162 CFIS96 44404418 Ki > 50 nM T67162 C36EZX 44404422 Ki = 29 nM T67162 CW4E0R 44404423 Ki = 12 nM T67162 CM6JK9 44404428 Ki = 12 nM T67162 C1CFY7 44404437 Ki = 21 nM T67162 CPL38O 44404439 Ki = 15 nM T67162 CAH1M6 44404440 Ki = 73 nM T67162 CC7DU3 44404443 Ki = 81 nM T67162 CAS49R 44404446 Ki > 100 nM T67162 C4I7RN 44404449 Ki = 11 nM T67162 CN6TX1 44404450 Ki = 92 nM T67162 C4HWE2 44404453 Ki = 35 nM T67162 C5ZV3O 44404454 Ki > 100 nM T67162 C34KQU 44404456 Ki > 100 nM T67162 C4NX6R 44404457 Ki = 59 nM T67162 C7SZ6O 44404459 Ki = 55 nM T67162 C01GEA 44404460 Ki = 16 nM T67162 C92LED 44404463 Ki = 17 nM T67162 C20AJE 44404465 Ki = 11 nM T67162 C2L7DW 44404470 Ki = 4 nM T67162 CQU19N 44405414 Ki = 38000 nM T67162 CJ3ED5 44405445 Ki = 500 nM T67162 CT5IP4 44405452 Ki = 29000 nM T67162 C9YLW2 44405455 Ki = 18000 nM T67162 C9Q7CS 44405466 Ki = 4460 nM T67162 CCP9V7 44405469 Ki = 230 nM T67162 CX7ER9 44405490 Ki = 1300 nM T67162 C3I8EC 44405492 Ki = 60 nM T67162 CD29AT 44405522 Ki = 1800 nM T67162 CF4S3Y 44405965 Ki = 137.2 nM T67162 CT3Z8U 44405980 Ki = 363.2 nM T67162 C0BI5F 44405985 Ki = 356.1 nM T67162 C4NC8M 44405995 Ki = 626.5 nM T67162 C0R5VL 44406003 Ki = 1720 nM T67162 CL5C9T 44406077 Ki = 164.6 nM T67162 CO2H3T 44406799 Ki > 10000 nM T67162 CI70SN 44406862 Ki > 10000 nM T67162 C0R6PK 44406863 Ki > 10000 nM T67162 CDA3R0 44406866 Ki > 10000 nM T67162 CU52FA 44406881 Ki > 10000 nM T67162 CRQ1J7 44406885 Ki = 82.1 nM T67162 COL64Y 44406886 Ki = 89.4 nM T67162 CSJ95I 44406895 Ki = 220 nM T67162 C0NHR2 44406899 Ki = 646 nM T67162 CT57XV 44406913 Ki = 148 nM T67162 CV8YF1 44406926 Ki = 302 nM T67162 CVU15M 44406983 Ki = 155 nM T67162 CPE1L4 44406984 Ki = 273 nM T67162 CH8L2V 44407007 Ki = 290 nM T67162 C0EXA1 44407083 IC50 > 10000 nM T67162 C8WD1P 44407270 Ki = 126 nM T67162 CDG04R 44407298 Ki = 669 nM T67162 C16HAY 44407300 Ki = 261 nM T67162 CVK80E 44407307 Ki = 289 nM T67162 C5HYM0 44407308 Ki = 354 nM T67162 C8VHO1 44407320 Ki = 254 nM T67162 C8QXI0 44407346 Ki = 467 nM T67162 CN52HW 44407347 Ki = 65 nM T67162 CCS63V 44407363 Ki = 93 nM T67162 C3V5TA 44407424 Ki = 243 nM T67162 C8SA0E 44407425 Ki = 151 nM T67162 CA64GU 44407436 Ki = 118 nM T67162 C74XRS 44407437 Ki = 83 nM T67162 CZ24HP 44408818 Ki = 0.55 nM T67162 C7AC1M 44409606 Ki = 231 nM T67162 C12HNJ 44409613 Ki = 137 nM T67162 C5A8GN 44409704 Ki = 409 nM T67162 CV9HI5 44409706 Ki = 212 nM T67162 C1AMJ7 44409707 Ki = 174 nM T67162 C9HR5I 44409720 Ki = 527 nM T67162 CR7XG9 44409721 Ki = 168 nM T67162 CDXJ02 44409726 Ki = 171 nM T67162 CKMT45 44409727 Ki = 234 nM T67162 CJ6LU7 44409730 Ki = 159 nM T67162 C4G9ZY 44409731 Ki = 17.3 nM T67162 CDW31B 44409888 Ki = 195 nM T67162 C31CNO 44409890 Ki = 65.8 nM T67162 C8V2XC 44409891 Ki = 91.3 nM T67162 CL26QH 44409908 Ki = 244 nM T67162 CP81TR 44409911 Ki = 59.1 nM T67162 C0VZ1B 44409913 Ki = 399 nM T67162 CJD14X 44409925 Ki = 128 nM T67162 CAO78Q 44411663 Ki > 1000 nM T67162 C8NVH0 44411664 Ki > 1000 nM T67162 C2Y8VK 44411667 Ki > 1000 nM T67162 C38VWG 44411668 Ki > 1000 nM T67162 C5Z2IY 44411674 Ki > 1000 nM T67162 CU2EY5 44411847 Ki > 1000 nM T67162 CD0OH1 44411864 Ki > 1000 nM T67162 CTLN43 44411929 Ki > 1000 nM T67162 CKX6D2 44411930 Ki > 1000 nM T67162 CQ89KF 44411933 Ki > 1000 nM T67162 CCJ1S9 44411934 Ki > 1000 nM T67162 CL28ZA 44411935 Ki > 1000 nM T67162 CG13DQ 44411936 Ki > 1000 nM T67162 CR2CJ9 44412182 Ki = 43 nM T67162 CF9IW1 44412191 Ki = 250 nM T67162 C8FU9P 44412268 Ki = 860 nM T67162 C78RSG 44412269 Ki = 65 nM T67162 CKY57Q 44412458 Ki = 110 nM T67162 CK9FC8 44412468 Ki = 190 nM T67162 C63XKI 44412482 Ki = 31 nM T67162 C2UBR0 44412494 Ki = 1900 nM T67162 CMO83R 44414898 EC50 > 10000 nM T67162 C4F1YB 44415054 EC50 > 10000 nM T67162 CW35JZ 44415055 EC50 > 10000 nM T67162 CMW2Z8 44415338 Ki = 2084 nM T67162 CQM07I 44415345 Ki > 3000 nM T67162 C5O7LC 44415367 Ki = 400 nM T67162 C8YWJ4 44415368 Ki = 1950 nM T67162 CX8TH3 44415382 Ki = 621 nM T67162 CS27IO 44415383 Ki = 582 nM T67162 CS6D0A 44415394 Ki = 1600 nM T67162 CO1L6U 44415473 Ki = 1900 nM T67162 C35IJK 44415506 Ki = 517 nM T67162 CK50IL 44415507 Ki = 1126 nM T67162 CQ57GR 44415517 Ki = 921 nM T67162 C4VWS0 44415518 Ki = 181 nM T67162 C8R3VX 44415535 Ki = 1776 nM T67162 CZ0RO7 44415536 Ki = 350 nM T67162 C98EFJ 44415543 Ki = 1150 nM T67162 C75DUR 44415544 Ki = 2386 nM T67162 C6I8EF 44415551 Ki = 9251 nM T67162 C3QAZ4 44415552 Ki = 1521 nM T67162 C69NUI 44415558 Ki = 931 nM T67162 CDP0Y7 44415560 Ki = 431 nM T67162 C0MFJ2 44415567 Ki = 3648 nM T67162 C58WLD 44415568 Ki = 1362 nM T67162 CU2FG6 44415569 Ki = 340 nM T67162 C7RU3M 44415577 Ki = 460 nM T67162 CIR8U5 44415578 Ki = 630 nM T67162 CC2PQ3 44415579 Ki = 3818 nM T67162 CD4CA5 44415582 Ki = 4927 nM T67162 CF90AU 44415584 Ki = 792 nM T67162 CDU6Y5 44415593 Ki = 458 nM T67162 C32GAH 44415594 Ki = 1314 nM T67162 CWQ9G5 44415595 Ki = 215 nM T67162 C38COL 44415598 Ki = 338 nM T67162 COT4H5 44415599 Ki = 63 nM T67162 CUQ7W3 44415600 Ki = 202 nM T67162 CR89VA 44415601 Ki = 533 nM T67162 C3M4HU 44415605 Ki = 1186 nM T67162 CFIT89 44415606 Ki = 1379 nM T67162 CHQ92K 44415611 Ki = 837 nM T67162 C9U7DG 44415612 Ki = 274 nM T67162 C1TYG7 44415613 Ki = 3772 nM T67162 CEO41K 44415615 Ki = 1126 nM T67162 C8O5AW 44415622 Ki > 3000 nM T67162 CW91OY 44415623 Ki > 2000 nM T67162 CB9XC7 44415624 Ki = 421 nM T67162 CA3JN6 44415625 Ki = 759 nM T67162 CM5WN1 44415628 Ki = 1474 nM T67162 CM2L3X 44415629 Ki = 2997 nM T67162 CMT3S0 44415633 Ki = 97 nM T67162 C2I8XJ 44415638 Ki > 2000 nM T67162 C64PWA 44415644 Ki > 3000 nM T67162 CIX23C 44415645 Ki > 2000 nM T67162 C6PMV8 44415646 Ki > 3000 nM T67162 CCM42T 44415647 Ki > 3000 nM T67162 CVZH14 44415648 Ki = 1261 nM T67162 C1MC3X 44415649 Ki = 3230 nM T67162 C3GVI9 44415657 Ki = 180 nM T67162 C9NQ4B 44415658 Ki = 78 nM T67162 C4YT5G 44415670 Ki = 69 nM T67162 CH0BY5 44415672 Ki = 383 nM T67162 C1SQ8J 44415673 Ki = 196 nM T67162 CM84OB 44415685 Ki = 270 nM T67162 CY69CA 44415686 Ki = 286 nM T67162 CZ76OD 44415688 Ki = 374 nM T67162 CK59CO 44415689 Ki = 496 nM T67162 C7AZ5D 44415690 Ki = 287 nM T67162 CRJ9N4 44415701 Ki = 267 nM T67162 C0D4BL 44415702 Ki = 175 nM T67162 CAR0F2 44415703 Ki = 6394 nM T67162 CEVY54 44415704 Ki = 1015 nM T67162 C1MC6P 44415705 Ki = 92 nM T67162 C3KG7M 44415721 Ki = 36 nM T67162 C1XRF4 44415723 Ki = 240 nM T67162 C0R4OV 44415724 Ki = 390 nM T67162 CL4W5C 44415738 Ki = 3896 nM T67162 CVS38E 44415743 Ki = 1969 nM T67162 C8BU4E 44415745 Ki = 608 nM T67162 C3AWV2 44415758 Ki > 3000 nM T67162 CH4O7P 44415759 Ki > 3000 nM T67162 CK5C8A 44415786 Ki > 3000 nM T67162 CQ5SV8 44415802 Ki = 828 nM T67162 CBMU18 44415804 Ki = 12710 nM T67162 CK76UE 44415805 Ki > 3000 nM T67162 C2S0MB 44415807 Ki = 1571 nM T67162 C5EO4H 44415822 Ki = 1616 nM T67162 CLY4R7 44415823 Ki = 28425 nM T67162 CEP25B 44415824 Ki = 709 nM T67162 C95DPW 44415825 Ki > 2000 nM T67162 CI5MF1 44415826 Ki = 231 nM T67162 C8JE2L 44415827 Ki = 197 nM T67162 CL0K9A 44415835 Ki = 5561 nM T67162 C5ELF8 44415836 Ki = 409 nM T67162 CPE3D9 44415837 Ki = 998 nM T67162 C8D9WN 44415838 Ki = 194 nM T67162 C7IR4G 44415839 Ki = 175 nM T67162 C2V6LX 44415844 Ki = 484 nM T67162 C2KG8A 44415845 Ki = 3000 nM T67162 C8I7FQ 44415848 Ki = 1280 nM T67162 CMC2Z1 44415849 Ki = 139 nM T67162 CNUD41 44415954 Ki = 1850 nM T67162 C89HPL 44417647 Ki = 340 nM T67162 CCPO37 44419053 Ki = 407.38 nM T67162 CGL9E1 44419056 Ki = 199.53 nM T67162 CP5M3H 44419060 Ki = 128.82 nM T67162 CJ4EZ9 44419065 Ki = 38.02 nM T67162 CIWX27 44419066 Ki = 218.78 nM T67162 CE2V0S 44425698 Ki = 794.33 nM T67162 C2TE3S 44425699 Ki = 199.53 nM T67162 C90AOQ 44425700 Ki = 398.11 nM T67162 CU52GB 44425701 Ki = 31.62 nM T67162 C9F1XP 44425702 Ki = 50.12 nM T67162 CR1QN5 44425703 Ki = 501.19 nM T67162 C5UZS7 44425704 Ki = 316.23 nM T67162 CN96FA 44425705 Ki = 100 nM T67162 C1J9MY 44425706 Ki = 15.85 nM T67162 CPI52U 44425708 Ki = 100 nM T67162 CNZ3M7 44425711 Ki = 63.1 nM T67162 C92AZG 44425714 Ki = 39.81 nM T67162 C7LP1B 44425717 Ki = 6.31 nM T67162 CX8TR0 44425719 Ki = 50.12 nM T67162 C7C4QE 44426404 Ki = 66 nM T67162 CE3XQ2 44426405 Ki = 104 nM T67162 CJN6P4 44427818 Ki = 28.3 nM T67162 CW3F5H 44427820 Ki = 23.6 nM T67162 CYLO03 44427821 Ki = 105 nM T67162 CJY9L5 44427822 Ki = 92 nM T67162 CO46HS 44427823 IC50 = 22.9 nM T67162 CFG0S3 44427824 Ki = 1160 nM T67162 C7PK0M 44427825 Ki = 69 nM T67162 CDV6A3 44427826 Ki = 48.4 nM T67162 C65ZXC 44427827 EC50 = 15.8 nM T67162 CZ0X7U 44427829 Ki = 319 nM T67162 C9U8YT 44427831 Ki = 284 nM T67162 C0C8AH 44427835 Ki = 134 nM T67162 C8EV3G 44427836 Ki = 28.4 nM T67162 CA96WP 44427839 Ki = 84 nM T67162 C46BRT 44427840 Ki = 68.4 nM T67162 CS9ND5 44427841 Ki = 53.7 nM T67162 COV6N3 44427842 Ki = 1050 nM T67162 CY0QJ2 44427970 Ki = 1028 nM T67162 CCRH08 44428207 Ki = 1258.93 nM T67162 C4G7QF 44431545 Ki = 34 nM T67162 C8OP5V 44431546 Ki = 2.4 nM T67162 C0B5TC 44431547 Ki = 31 nM T67162 CCXB24 44431548 Ki = 51 nM T67162 C5QI0V 44431551 Ki = 64 nM T67162 C2R4TP 44431553 Ki = 39 nM T67162 COIS42 44431554 Ki = 27 nM T67162 C0APQ4 44431555 Ki = 14 nM T67162 CJT34W 44431557 Ki = 58 nM T67162 CF76RP 44431560 Ki = 62 nM T67162 CY8C0V 44431562 Ki = 62 nM T67162 C2UD6M 44431564 Ki = 50 nM T67162 C4J0TG 44431574 Ki = 139 nM T67162 C0C8TU 44431587 Ki = 36 nM T67162 C1QV6S 44431590 Ki = 1.9 nM T67162 CF3ST7 44431594 Ki = 18 nM T67162 CA9O2E 44431599 Ki = 52 nM T67162 CX9YA2 44431602 Ki = 42 nM T67162 C9OSE8 44431607 Ki = 198 nM T67162 CT0LP1 44431611 Ki = 42 nM T67162 C46NHX 44431612 Ki = 356 nM T67162 C3IA4W 44431613 Ki = 123 nM T67162 C5QJ8S 44431614 Ki = 588 nM T67162 CXD1Q9 44431615 Ki = 425 nM T67162 C0WPS6 44431616 Ki = 24 nM T67162 C4SZA3 44431617 Ki = 15 nM T67162 CE6L0D 44431618 Ki = 43 nM T67162 CS9N3Q 44431620 Ki = 61 nM T67162 CEWQ41 44433348 Ki = 2.7 nM T67162 C2AZ6B 44436300 Ki = 4.1 nM T67162 C30QMX 44436301 Ki = 177 nM T67162 C9AJ0D 44436302 Ki = 6.2 nM T67162 C3NVL0 44436303 Ki = 46 nM T67162 CREM27 44436304 Ki = 140 nM T67162 C53XYK 44436305 Ki = 73 nM T67162 C2LF9K 44436306 Ki = 323 nM T67162 C9H8ST 44436307 Ki = 760 nM T67162 C7IBE2 44436308 Ki = 26 nM T67162 C2B4WN 44436596 Ki = 48 nM T67162 CLV2E1 44436597 Ki = 4700 nM T67162 C0LBO6 44436598 Ki = 83 nM T67162 CREV94 44436599 Ki = 1200 nM T67162 CZ37MU 44436600 Ki = 160 nM T67162 CRW39P 44436601 Ki = 190 nM T67162 CG06FU 44436602 Ki = 78 nM T67162 C2GD0Z 44436603 Ki = 280 nM T67162 C1T9IF 44436605 Ki = 15 nM T67162 CBQ6F7 44436606 Ki = 780 nM T67162 C6ZJ1W 44436608 Ki = 15 nM T67162 C1OP6H 44436610 Ki = 210 nM T67162 CR6UK2 44436617 Ki = 27 nM T67162 CHTG80 44436618 Ki = 11 nM T67162 CI5K6A 44436621 Ki = 23 nM T67162 CW7VF4 44436719 Ki = 1180 nM T67162 CP85SY 44436720 Ki = 226 nM T67162 C1J6BZ 44436721 Ki = 457 nM T67162 C8I7HR 44436722 Ki = 590 nM T67162 CLU0F7 44436723 Ki = 621 nM T67162 CE0M4N 44436724 Ki = 435 nM T67162 CR7Y8E 44436725 Ki = 587 nM T67162 CFP41N 44436726 Ki = 963 nM T67162 C7QH5X 44436727 Ki = 1000 nM T67162 C04VDB 44436728 Ki = 160 nM T67162 C4ZN9T 44436729 Ki = 189 nM T67162 C2V4IE 44436730 Ki = 136 nM T67162 C4ZN9E 44436731 Ki = 161 nM T67162 C29BYE 44436732 Ki = 633 nM T67162 C6UWG1 44436735 Ki = 663 nM T67162 C4GX5V 44436737 Ki = 626 nM T67162 C9YC8V 44436739 Ki = 313 nM T67162 CDT72W 44436741 Ki = 972 nM T67162 C1J2MR 44436743 Ki = 619 nM T67162 C4HR8W 44436745 Ki = 1324 nM T67162 CZ6H2Q 44436746 Ki = 429 nM T67162 CAD4I1 44436747 Ki = 4925 nM T67162 C8PX3T 44436748 Ki = 497 nM T67162 C8BO7G 44436750 Ki = 258 nM T67162 C5L3JM 44436751 Ki = 1149 nM T67162 CXI70P 44436753 Ki > 1000 nM T67162 CGP8C7 44436756 Ki = 252 nM T67162 C6K9DT 44436759 Ki = 849 nM T67162 CCL5K1 44436762 Ki = 128 nM T67162 CZ5V0R 44436765 Ki = 1570 nM T67162 C7Y5VG 44436767 Ki = 13350 nM T67162 CN49HQ 44436768 Ki > 1000 nM T67162 C06RTZ 44436769 Ki = 4620 nM T67162 C6JQ1H 44436771 Ki = 163 nM T67162 CN2Q5J 44436772 Ki > 1000 nM T67162 CG2X1D 44437896 Ki = 14 nM T67162 CX04CK 44437897 Ki = 23 nM T67162 CC4V7G 44438186 Ki = 382 nM T67162 CJ8W5C 44438197 Ki = 26.1 nM T67162 CMGT04 44438199 EC50 = 83.4 nM T67162 C8C0HP 44438201 Ki = 6.9 nM T67162 CJDT47 44438203 EC50 = 69.1 nM T67162 CU4AS8 44438204 Ki = 127 nM T67162 CPAE72 44438206 Ki = 5360 nM T67162 CJM3K5 44438208 Ki = 177 nM T67162 CPH7V5 44438209 Ki = 159 nM T67162 C6K3ZU 44438210 Ki = 98.4 nM T67162 CADG24 44438211 Ki = 201 nM T67162 CLE5G1 44438213 Ki = 2890 nM T67162 C8ILG5 44438215 Ki = 4265 nM T67162 CFE50G 44438218 EC50 = 314 nM T67162 C3KS0B 44438219 Ki = 184 nM T67162 CAQ5Y9 44438220 EC50 = 24.8 nM T67162 C52KTZ 44438221 Ki = 120 nM T67162 C8LW2C 44438222 Ki = 199 nM T67162 CF2WK6 44438223 Ki = 60 nM T67162 CVT06Y 44438224 Ki = 58.8 nM T67162 C4POI0 44438225 Ki > 10000 nM T67162 CO76KJ 44438226 Ki = 2000 nM T67162 CJZ69F 44438227 Ki = 2370 nM T67162 CS1H8X 44438228 EC50 = 34.7 nM T67162 CEQ1L8 44438229 Ki = 165 nM T67162 CUF21H 44438230 EC50 = 2.13 nM T67162 CU49FT 44438231 Ki = 438 nM T67162 CD89OH 44438232 Ki = 548 nM T67162 C0VA9W 44438233 Ki = 21 nM T67162 CJSX04 44438234 Ki = 21 nM T67162 CWE9K4 44438235 Ki = 54 nM T67162 C5Q6PG 44438236 EC50 = 20 nM T67162 CWS8R5 44438237 EC50 = 166 nM T67162 C4BJ9F 44438238 Ki > 10000 nM T67162 CL4FV8 44438239 Ki = 23.9 nM T67162 CKZF16 44439165 Ki = 3162.28 nM T67162 CA4HZ3 44439167 Ki = 2511.89 nM T67162 CQ18PR 44439374 Ki > 1000 nM T67162 CN9RH5 44439375 Ki > 1000 nM T67162 C2X1FS 44439377 Ki > 2000 nM T67162 CW2KQ1 44439378 Ki > 2000 nM T67162 C2J9LG 44439379 Ki > 2000 nM T67162 COKH57 44439380 Ki > 2000 nM T67162 CO20GU 44439381 Ki > 2000 nM T67162 C4KQ8C 44439384 Ki > 2000 nM T67162 CQXS03 44439385 Ki > 2000 nM T67162 CRC2Y5 44439387 Ki = 31000 nM T67162 C3ZT7I 44439388 Ki = 25000 nM T67162 CKU9N8 44439389 Ki = 200000 nM T67162 C20VDP 44439390 Ki = 1500 nM T67162 C6RKA9 44439391 Ki = 1900 nM T67162 CPX5Q2 44439396 Ki = 2400 nM T67162 C2R0SX 44439397 Ki = 54000 nM T67162 C4CMV7 44439398 Ki = 11000 nM T67162 C8YQ4P 44439399 Ki = 14000 nM T67162 C6YA9O 44439400 Ki = 42000 nM T67162 C89ZPX 44439401 Ki = 14000 nM T67162 CE60JL 44439402 Ki > 300000 nM T67162 C65GSE 44439403 Ki = 12000 nM T67162 CKUG90 44439404 Ki = 1700 nM T67162 CTYP87 44439405 Ki > 100000 nM T67162 C3UBA6 44439406 Ki = 8200 nM T67162 C7HV8X 44439407 Ki = 3100 nM T67162 CD4T3S 44439408 Ki > 100000 nM T67162 C07XPE 44439409 Ki = 1600 nM T67162 CMU43Q 44439410 Ki = 59000 nM T67162 CBI86V 44439942 Ki = 11.9 nM T67162 C3HMI2 44439943 Ki = 38.4 nM T67162 C63PQV 44439944 Ki = 22.8 nM T67162 C2P4CI 44439945 Ki = 74.7 nM T67162 C3OD9X 44441217 Ki < 398.11 nM T67162 CY29KE 44441218 Ki < 10000 nM T67162 CRPB21 44441219 Ki < 10000 nM T67162 C6JU0E 44441222 Ki < 10000 nM T67162 CG4SU7 44441225 Ki < 120.23 nM T67162 C1UAM5 44443901 EC50 = 7200 nM T67162 CU96SV 44443902 EC50 > 30000 nM T67162 CIJ85M 44443903 EC50 > 100000 nM T67162 CZ34PG 44443904 EC50 > 10000 nM T67162 C4BUQ3 44443905 EC50 > 10000 nM T67162 CS21LM 44443907 EC50 > 1000 nM T67162 CQ27IL 44443908 EC50 > 10000 nM T67162 CBL7R2 44443909 EC50 > 10000 nM T67162 C8KWH4 44443911 EC50 > 10000 nM T67162 CGM1A8 44443915 EC50 > 1000 nM T67162 CV06CS 44443916 EC50 > 1000 nM T67162 CF15SI 44443920 EC50 > 10000 nM T67162 C5RVE0 44446999 Ki = 10 nM T67162 C9E0FL 44447001 Ki = 21 nM T67162 CSJ4U5 44447002 Ki = 34 nM T67162 CL87PU 44447003 Ki = 27 nM T67162 CCD6B5 44447005 Ki = 21 nM T67162 CBH65G 44447007 Ki = 67 nM T67162 C8CF7X 44447008 Ki = 22 nM T67162 CN3EH7 44447010 Ki = 15 nM T67162 CYWP06 44447012 Ki = 5 nM T67162 C41KNM 44447013 Ki = 6 nM T67162 CE12BC 44447015 Ki = 6 nM T67162 CUD31L 44447018 Ki = 26 nM T67162 CNLX79 44447028 Ki = 33 nM T67162 CM8K1H 44447039 Ki = 5 nM T67162 C5IJW2 44447059 Ki = 3 nM T67162 CHXF10 44447061 Ki = 8 nM T67162 CM8P9A 44447070 Ki = 10 nM T67162 CK4HA6 44447072 Ki = 5 nM T67162 C2S6HQ 44448054 Ki = 6110 nM T67162 C3Z7FI 44451927 IC50 = 5300 nM T67162 C57SBC 44451980 IC50 = 140 nM T67162 CEST18 44451982 IC50 = 4000 nM T67162 CRN4F8 44452007 IC50 = 1500 nM T67162 CG1C6X 44452142 IC50 = 6600 nM T67162 CVAU93 44452222 IC50 = 6900 nM T67162 C0B3LC 44452327 IC50 = 1500 nM T67162 CB1MX2 44454118 Ki > 2511.89 nM T67162 CR3IC6 44454120 Ki > 2511.89 nM T67162 C5B0IF 44454150 Ki < 630.96 nM T67162 CRD82N 44454166 Ki > 1000 nM T67162 CMVS90 44454167 Ki > 630.96 nM T67162 C7FY1E 44454168 Ki > 1258.93 nM T67162 CW4S3P 44454190 Ki = 316.23 nM T67162 C7H3CL 44454192 Ki > 1000 nM T67162 CU0N1E 44454217 Ki > 1584.89 nM T67162 C9DBA3 44454218 Ki > 1000 nM T67162 CK01QH 44454219 Ki > 1000 nM T67162 CLO6X0 44454223 Ki > 2511.89 nM T67162 CECR53 44454247 Ki > 794.33 nM T67162 CD4ZU7 44454248 Ki > 1000 nM T67162 CS2N1D 44454275 Ki > 1000 nM T67162 CJ5XB1 44454278 Ki > 10000 nM T67162 C4GON0 44454309 Ki > 2511.89 nM T67162 C91PHS 44454318 Ki < 794.33 nM T67162 CT50UC 44454320 Ki < 794.33 nM T67162 C35WYK 44454339 Ki > 1000 nM T67162 CZO96M 44454340 Ki > 1000 nM T67162 C2CIO7 44454351 Ki < 794.33 nM T67162 C9AH1O 44454352 Ki < 794.33 nM T67162 CM8H2G 44454353 Ki < 1258.93 nM T67162 C1EZP7 44454358 Ki < 501.19 nM T67162 CEB84V 44454371 Ki > 794.33 nM T67162 C5EV7Z 44454381 Ki < 1258.93 nM T67162 CWC92Y 44454382 Ki < 1258.93 nM T67162 CH0S2F 44454384 Ki < 1258.93 nM T67162 C32LHE 44454400 Ki > 1000 nM T67162 CG18KC 44454401 Ki > 1000 nM T67162 CI0CJ9 44454402 Ki > 630.96 nM T67162 CP34QH 44454403 Ki > 630.96 nM T67162 CW4OX5 44454418 Ki < 398.11 nM T67162 CW1I4Z 44454420 Ki < 1000 nM T67162 C8TJW4 44454434 Ki > 1000 nM T67162 CX9U8I 44454443 Ki < 794.33 nM T67162 CXA7W2 44454458 Ki > 630.96 nM T67162 CBGJ08 44454459 Ki > 630.96 nM T67162 CB1P9X 44454685 Ki = 590 nM T67162 CZJ8G6 44454707 Ki = 1100 nM T67162 CC5SL3 44454709 Ki = 94 nM T67162 CD6M2F 44454710 Ki = 21000 nM T67162 C5V3RI 44454711 Ki = 57 nM T67162 C1GKA2 44454734 Ki = 120 nM T67162 CBD62A 44454735 Ki = 310 nM T67162 CZL97F 44455426 Ki > 10000 nM T67162 C12XGE 44456400 Ki > 10000 nM T67162 CO6L0A 44457584 Ki = 630 nM T67162 CS14UN 44457651 Ki = 57 nM T67162 CLFG23 44457652 Ki = 800 nM T67162 CL1F7V 44459452 Ki = 310 nM T67162 CF8DR7 44459463 Ki = 90 nM T67162 C86HXK 44460799 IC50 > 1000 nM T67162 CQ2IX7 44461606 IC50 = 9549.93 nM T67162 C4DL5C 44469677 IC50 > 10000 nM T67162 CWPH50 44478261 Ki = 328 nM T67162 C9OY3U 44517726 Ki = 100 nM T67162 C8C3UM 44533248 Ki = 125.89 nM T67162 C4SX7H 44537919 Ki = 19.1 nM T67162 CVD14L 44537925 Ki = 80 nM T67162 C3D4HR 44537940 Ki = 605 nM T67162 CJ7U3K 44554227 Ki = 2036 nM T67162 CM0I1P 44554393 Ki = 1903 nM T67162 CNHA47 44554395 Ki = 2243 nM T67162 CRJ2I6 44554468 EC50 = 0.8 nM T67162 CX4D1K 44554470 EC50 = 4 nM T67162 CYL5M9 44554472 EC50 = 0.14 nM T67162 C8F9OM 44554474 EC50 = 1.1 nM T67162 CLZ37T 44554643 EC50 = 18 nM T67162 CV65YO 44554644 EC50 = 1400 nM T67162 CK2Y5P 44554649 EC50 = 0.5 nM T67162 C1MT5G 44554818 EC50 = 1.7 nM T67162 CQ1C7K 44554820 EC50 = 0.6 nM T67162 C7Z5IX 44554982 EC50 = 1.5 nM T67162 C7EI4P 44554984 EC50 = 1 nM T67162 CA3M1E 44554986 EC50 = 2.1 nM T67162 C7B4VN 44554987 EC50 = 3.5 nM T67162 CIZ2A5 44555137 EC50 = 13 nM T67162 CQ8JA9 44555138 EC50 = 33 nM T67162 C16HEZ 44555445 Ki > 10000 nM T67162 CJSC58 44561317 Ki = 77.62 nM T67162 C5SP0Z 44578445 Ki = 155 nM T67162 CVR7A5 44578446 Ki = 170 nM T67162 CXV4U0 44578885 Ki > 10000 nM T67162 CCIT12 44578976 IC50 = 1130 nM T67162 CST84W 44579032 Ki > 10000 nM T67162 CV32GO 44579033 Ki > 10000 nM T67162 C61JVZ 44579034 Ki > 10000 nM T67162 C2DFV7 44579418 IC50 > 10000 nM T67162 CTC8H6 44579419 IC50 > 10000 nM T67162 CYR0O3 44579457 IC50 = 2690 nM T67162 CF1EA4 44579458 IC50 > 10000 nM T67162 C49LWN 44579621 Ki > 10000 nM T67162 CZ6AK4 44579622 Ki > 10000 nM T67162 C5NS6H 44581972 Ki = 5248.07 nM T67162 CK8Z1P 44581973 Ki = 4897.79 nM T67162 C3UQ9Z 44581974 Ki = 5128.61 nM T67162 C21GPX 44582115 Ki = 11.48 nM T67162 CQEF30 44582140 Ki = 158.49 nM T67162 CVE23P 44582178 Ki = 229.09 nM T67162 COZ2M5 44582179 Ki = 151.36 nM T67162 CS7P4T 44582187 Ki = 20.42 nM T67162 CLHG02 44582491 Ki = 794.33 nM T67162 CN53TE 44582492 Ki > 100000 nM T67162 CZK49H 44582518 Ki = 218.78 nM T67162 CRCH48 44582675 Ki = 2686 nM T67162 CEJ4R8 44582676 Ki = 3828 nM T67162 C5QB4K 44582678 Ki > 10000 nM T67162 C01RCI 44582705 Ki > 10000 nM T67162 CXK14L 44586762 IC50 = 17.1 nM T67162 CFW0V8 44589129 Ki = 89.4 nM T67162 CCJK60 44589130 Ki = 243 nM T67162 C8GY9A 44589131 Ki > 100 nM T67162 CZ8VE0 44589175 Ki = 121 nM T67162 C2C7LE 44589176 Ki > 100 nM T67162 CYF42C 44589177 Ki > 100 nM T67162 C08TSZ 44589178 Ki = 17.8 nM T67162 C6VA9C 44589179 Ki = 196 nM T67162 C0LDK7 44589180 Ki > 100 nM T67162 CFB81M 44589377 Ki = 133 nM T67162 CS0QD1 44589378 Ki = 1341 nM T67162 CL40CM 44589593 IC50 > 10000 nM T67162 CKS5V4 44589594 IC50 = 3600 nM T67162 CXB30W 44589595 IC50 > 10000 nM T67162 CM5LJ8 44589596 IC50 = 2300 nM T67162 CPXE19 44589643 IC50 = 2700 nM T67162 C8AJO6 44589644 IC50 = 1100 nM T67162 CFS1A4 44589645 IC50 = 1900 nM T67162 C71EHI 44589646 IC50 > 10000 nM T67162 CP6ZA9 44591012 Ki = 904 nM T67162 C8S1HM 44591042 Ki = 53 nM T67162 C5C6GE 44591045 Ki = 970 nM T67162 C4YRD3 44591086 Ki = 588 nM T67162 CS5Q7A 44591087 Ki > 10000 nM T67162 CPA4R6 44591088 Ki = 170 nM T67162 CU37BO 44591098 Ki > 1000 nM T67162 CU48CL 44591099 Ki = 101 nM T67162 C7H9SE 44591134 Ki = 41 nM T67162 C6RLW0 44591135 Ki = 52 nM T67162 CBXW20 44591540 Ki > 10000 nM T67162 CSO48Z 44591564 Ki > 1000 nM T67162 CYV0C8 44591565 Ki > 10000 nM T67162 CH42OK 44591566 Ki > 10000 nM T67162 CT4LV3 44591587 Ki = 4570.88 nM T67162 C8AY3N 44591605 Ki > 10000 nM T67162 C67KZG 44608359 IC50 = 9.1 nM T67162 C8M2WP 44621617 EC50 = 0.6457 nM T67162 CU3LE6 44626329 Ki = 17 nM T67162 C9N4MQ 44626527 Ki = 398.11 nM T67162 CSJ9F1 44626530 Ki = 19.95 nM T67162 CCLQ67 44626632 Ki = 158.49 nM T67162 CA93OY 44626637 Ki = 316.23 nM T67162 CPML65 44626639 Ki = 3981.07 nM T67162 CDA90T 44626641 Ki = 6309.57 nM T67162 C2TBL0 44626734 Ki = 398.11 nM T67162 C7LUV5 44626738 Ki > 398.11 nM T67162 CRCL97 44626740 Ki = 199.53 nM T67162 CZ25SY 44626744 Ki = 158.49 nM T67162 C5DM7T 44626835 Ki > 794.33 nM T67162 C85ZIF 44626928 Ki > 1258.93 nM T67162 C4BYG5 44626929 Ki = 125.89 nM T67162 CK5BG2 44626935 Ki > 794.33 nM T67162 CWL84Q 44627022 Ki = 199.53 nM T67162 CGXJ71 44627023 Ki = 79.43 nM T67162 CBP18J 44627024 Ki > 1000 nM T67162 C30KEM 44627025 Ki = 125.89 nM T67162 CV1DO3 44627033 Ki = 125.89 nM T67162 CAH6O1 44627120 Ki = 100 nM T67162 CUE56O 44627123 Ki = 158.49 nM T67162 CDY32E 44627127 Ki = 50.12 nM T67162 CJ4ZQ0 44627129 Ki = 316.23 nM T67162 CN1O6P 44627131 Ki = 158.49 nM T67162 CQE59L 44627133 Ki = 31.62 nM T67162 C4QV9Y 44627238 Ki > 794.33 nM T67162 C1D5FJ 44627240 Ki = 158.49 nM T67162 CNK4P0 44627242 Ki = 12.59 nM T67162 CY3LE2 44627245 Ki > 1000 nM T67162 C5LN9E 44627351 Ki = 31.62 nM T67162 CLUN07 44627353 Ki = 158.49 nM T67162 CZ1FY5 44627355 Ki = 63.1 nM T67162 C3ZWA4 44627357 Ki = 79.43 nM T67162 CY1TE0 44627358 Ki > 398.11 nM T67162 CG97OK 44627359 Ki = 12.59 nM T67162 C65RAG 44627466 Ki > 630.96 nM T67162 C06TJC 44627468 Ki = 316.23 nM T67162 CBV8I6 44627470 Ki = 158.49 nM T67162 C6C9EI 45006130 Ki = 0.3236 nM T67162 CQI0D4 45102707 Ki > 794.33 nM T67162 CSEP-69 45102708 Ki > 3162.28 nM T67162 C0DLU3 45109862 IC50 = 1071 nM T67162 CQ7D5U 45140376 EC50 = 1.69 nM T67162 CSV08Y 45140377 Ki = 3.75 nM T67162 C98UOH 45260312 Ki = 1584.89 nM T67162 C6Y0LZ 45260341 Ki = 199.53 nM T67162 CHLR80 45260355 Ki = 794.33 nM T67162 C8F1MO 45260357 Ki = 794.33 nM T67162 C31CPA 45260363 Ki = 199.53 nM T67162 CNQ7G1 45260372 Ki = 158.49 nM T67162 C2YL4K 45260377 Ki = 630.96 nM T67162 CXMW87 45260407 Ki = 398.11 nM T67162 C7LRZ1 45260417 Ki = 316.23 nM T67162 CJ89IW 45260733 Ki = 1900 nM T67162 CG0BL7 45261538 Ki = 19 nM T67162 CW0X2M 45262323 Ki = 251.19 nM T67162 CQ58RZ 45262339 Ki = 199.53 nM T67162 CE6I0O 45262343 Ki = 125.89 nM T67162 CY87WP 45262345 Ki = 199.53 nM T67162 C6Y4HQ 45262347 Ki = 63.1 nM T67162 C24FEH 45262348 Ki = 316.23 nM T67162 CU03YK 45262349 Ki = 398.11 nM T67162 C3QCD6 45262363 Ki = 316.23 nM T67162 CAT04I 45262369 Ki = 158.49 nM T67162 CY3FD0 45262381 Ki = 79.43 nM T67162 C6PGT0 45262384 Ki = 125.89 nM T67162 C08TZA 45262385 Ki = 630.96 nM T67162 CNE0B7 45262402 Ki = 158.49 nM T67162 CQ29HI 45262403 Ki = 31.62 nM T67162 C4U7YW 45262404 Ki = 79.43 nM T67162 CF15EW 45262410 Ki = 501.19 nM T67162 CO0HX8 45262412 Ki = 125.89 nM T67162 C08KWJ 45262415 Ki = 251.19 nM T67162 C9FD2N 45262416 Ki = 630.96 nM T67162 CB6KO5 45262417 Ki = 630.96 nM T67162 C1Q9WD 45264008 Ki = 79.43 nM T67162 C4L3JP 45265219 Ki = 199.53 nM T67162 CR0N7U 45265240 Ki = 199.53 nM T67162 C2A3HT 45265244 Ki = 794.33 nM T67162 CR7UF5 45265257 Ki = 501.19 nM T67162 C5RW2P 45265266 Ki = 398.11 nM T67162 C7N2DT 45265305 Ki = 630.96 nM T67162 C4B6JW 45265589 Ki = 63.1 nM T67162 C52ALF 45265590 Ki = 316.23 nM T67162 CE2YT8 45265597 Ki = 199.53 nM T67162 CLVE65 45265605 Ki = 158.49 nM T67162 CEUN59 45265612 Ki = 100 nM T67162 C4QY5J 45265633 Ki = 316.23 nM T67162 CPR46X 45265656 Ki = 124.4 nM T67162 CAHW68 45267251 Ki = 158.49 nM T67162 CW1S6B 45267254 Ki = 100 nM T67162 CD47IO 45267261 Ki > 10000 nM T67162 CJPS81 45267262 Ki > 10000 nM T67162 C4HOR6 45267270 Ki = 25.12 nM T67162 CM2YT9 45267409 Ki = 40000 nM T67162 CCLR12 45267435 Ki = 2600 nM T67162 CPD18Y 45267471 Ki = 3.981 nM T67162 CL0WP4 45267480 Ki = 25.12 nM T67162 C2H4ZX 45267491 Ki = 3.162 nM T67162 C0KTX2 45267492 Ki = 316.23 nM T67162 C2R9HN 45267503 Ki = 1000 nM T67162 CEY87M 45267504 Ki = 251.19 nM T67162 CF2R3T 45268112 Ki = 6.31 nM T67162 C3S5ZP 45268113 Ki = 39.81 nM T67162 C0UG9Z 45268119 Ki = 158.49 nM T67162 C37TAV 45268120 Ki = 630.96 nM T67162 CP1TV2 45268127 Ki > 10000 nM T67162 C79VFY 45268141 Ki = 158.49 nM T67162 C64NZQ 45268142 Ki = 158.49 nM T67162 CENZ75 45268148 Ki = 199.53 nM T67162 C71SGH 45268292 Ki = 380 nM T67162 CL0CW7 45268293 Ki = 730 nM T67162 CM1SA7 45268333 Ki = 316.23 nM T67162 CH53XO 45268345 Ki = 251.19 nM T67162 CHB5U0 45268346 Ki = 501.19 nM T67162 COCN89 45268373 Ki = 1584.89 nM T67162 C4MU3C 45268438 Ki = 25.12 nM T67162 CEK21M 45268987 Ki = 794.33 nM T67162 CHB76Z 45268990 Ki = 316.23 nM T67162 CR3YU9 45268999 Ki > 10000 nM T67162 CW57CP 45269000 Ki = 1000 nM T67162 CYQ1I7 45269020 Ki = 12.59 nM T67162 C0F9UT 45269161 Ki = 10000 nM T67162 CQP0N3 45269168 Ki = 400 nM T67162 CVH8S4 45269235 Ki = 630.96 nM T67162 CU02ZQ 45269860 Ki = 398.11 nM T67162 CJ18ZC 45270021 Ki = 8600 nM T67162 CF43XE 45270678 Ki = 501.19 nM T67162 CK01NU 45270702 Ki > 10000 nM T67162 CL42RS 45270813 Ki = 160 nM T67162 C5RX4W 45270861 Ki = 3500 nM T67162 CO0P8H 45270903 Ki = 25.12 nM T67162 C7OM4D 45270916 Ki = 158.49 nM T67162 CMQ25P 45271491 Ki = 251.19 nM T67162 CEQ19M 45271499 Ki = 501.19 nM T67162 CESN63 45271510 Ki = 15.85 nM T67162 CMDC23 45271511 Ki = 39.81 nM T67162 C8TXI5 45271516 Ki = 1000 nM T67162 C5P3FX 45271520 Ki = 251.19 nM T67162 CF9I3G 45271548 Ki = 50.12 nM T67162 C4AJP5 45271653 Ki = 9100 nM T67162 C13RSZ 45271691 Ki = 26000 nM T67162 C6R3LQ 45271737 Ki = 100 nM T67162 CM5Q8S 45271738 Ki = 15.85 nM T67162 C42EJD 45271753 Ki = 100 nM T67162 CT3DP1 45271760 Ki = 50.12 nM T67162 C5U7LD 45272411 Ki > 10000 nM T67162 CM9W5B 45272412 Ki > 10000 nM T67162 CG9CO5 45272414 Ki = 251.19 nM T67162 C4W9NG 45272415 Ki = 794.33 nM T67162 C12WFN 45272425 Ki > 10000 nM T67162 CK67XC 45272426 Ki = 19.95 nM T67162 CQ2ZS6 45272434 Ki = 316.23 nM T67162 CGKZ21 45272435 Ki > 10000 nM T67162 CH0MA8 45272437 Ki = 2511.89 nM T67162 CW2MD0 45272438 Ki = 501.19 nM T67162 CZ8VO5 45272537 Ki = 2300 nM T67162 CGZW61 45272580 Ki = 570 nM T67162 CE1P8L 45272616 Ki = 31.62 nM T67162 CEO57P 45272634 Ki = 125.89 nM T67162 CI7C1L 45272635 Ki = 19.95 nM T67162 C9M6XP 45273045 Ki = 280 nM T67162 CIX32S 45273211 EC50 = 41.2 nM T67162 CX1QY9 45273266 Ki = 31.62 nM T67162 C62LGY 45273272 Ki = 251.19 nM T67162 CZ2OL1 45273273 Ki = 1258.93 nM T67162 C1YTJ8 45273278 Ki > 10000 nM T67162 CBM9R2 45273292 Ki = 100 nM T67162 CS04AC 45273293 Ki > 10000 nM T67162 CS95IU 45273334 Ki = 79.43 nM T67162 C19BMF 45273442 Ki = 3300 nM T67162 C7VR4A 45273443 Ki = 180 nM T67162 CFY94G 45273510 Ki = 79.43 nM T67162 CRSF80 45273522 Ki = 5.012 nM T67162 C3DB8P 45273523 Ki = 25.12 nM T67162 CM10UD 45273529 Ki = 79.43 nM T67162 CRD9C8 45273530 Ki = 50.12 nM T67162 CNQJ09 45273545 Ki = 125.89 nM T67162 C7XC3T 45273551 Ki = 199.53 nM T67162 CZ71RN 45278805 IC50 = 2542 nM T67162 CZN6M7 45278882 IC50 = 3736 nM T67162 CKQG15 45361874 Ki = 603 nM T67162 CYJ7P8 45379368 Ki > 10000 nM T67162 CU2CA7 45379369 Ki = 4 nM T67162 CT3K8Y 45379370 Ki = 55.1 nM T67162 CT3A1Q 45379373 Ki > 10000 nM T67162 C8TRE1 45379377 Ki = 4458 nM T67162 CML67J 45379515 Ki = 1476 nM T67162 C7MO3G 45481875 Ki = 39.1 nM T67162 C7S9HJ 45481888 Ki = 115 nM T67162 C0HPW1 45481889 Ki = 200 nM T67162 C0SF6L 45482151 Ki = 6.5 nM T67162 CXC65S 45482152 Ki = 17 nM T67162 C8TE2Y 45482153 Ki = 49 nM T67162 C9LX5P 45482169 Ki = 44 nM T67162 CJD2A3 45482180 Ki = 1 nM T67162 C0CHF4 45482789 IC50 = 1590 nM T67162 CQ9FN0 45483190 Ki = 33.88 nM T67162 CEZW26 45483246 Ki = 630.96 nM T67162 CLO70J 45483261 Ki = 158.49 nM T67162 C7LD5K 45483269 Ki = 32.36 nM T67162 CG5TR7 45483288 Ki = 234.42 nM T67162 CO1M6P 45483654 Ki = 10000 nM T67162 CIV3Q4 45483655 Ki = 770 nM T67162 C9D0RB 45486325 EC50 = 77.2 nM T67162 CD2OP0 45486328 EC50 = 13.5 nM T67162 C75KWB 45486329 Ki = 8.85 nM T67162 C41IVO 45486330 EC50 = 116 nM T67162 CPSV53 45486332 Ki = 7.08 nM T67162 C8NS2H 45486333 Ki = 270 nM T67162 C5BR3T 45486336 Ki = 5.22 nM T67162 CCVJ58 45486341 Ki = 21.7 nM T67162 CLK12R 45486360 Ki = 4.89 nM T67162 CU5LO4 45486363 Ki = 13.5 nM T67162 C9G1TW 45486364 Ki = 3.74 nM T67162 CA60OT 45486819 Ki = 50 nM T67162 CQMJ83 45486820 Ki = 12 nM T67162 CJN7X0 45486824 Ki = 3 nM T67162 CSIO35 45486825 Ki = 720 nM T67162 CFCD10 45486840 Ki = 24 nM T67162 C49EAG 45486845 Ki = 120 nM T67162 C6ROX8 45486859 Ki = 15 nM T67162 C6Q4AJ 45486879 Ki = 100 nM T67162 CY9ZD8 45486887 Ki = 36 nM T67162 C9BSL5 45486891 Ki = 45 nM T67162 CB0JM3 45486892 Ki = 220 nM T67162 CO9JN6 45486893 Ki = 140 nM T67162 CI8NA1 45486898 Ki = 310 nM T67162 C4H7OT 45486902 Ki = 28 nM T67162 CSQ1J5 45487336 Ki > 2511.89 nM T67162 C24WVU 45487513 Ki = 1584.89 nM T67162 C83MKA 45560581 Ki = 2300 nM T67162 CXT96Y 45815848 Ki > 10000 nM T67162 CV7C2M 45827434 Ki > 10000 nM T67162 C05PBD 46176231 Ki = 174 nM T67162 CI3WX2 46176232 Ki > 10000 nM T67162 C4XRY7 46176233 Ki = 342 nM T67162 C4WJ0Z 46176312 Ki = 296 nM T67162 CK9EC3 46180160 Ki = 3.74 nM T67162 C8YH5K 46180191 Ki > 10000 nM T67162 C5CET8 46180192 Ki > 10000 nM T67162 CEW06P 46180193 Ki > 10000 nM T67162 C9PBQ4 46180194 Ki > 10000 nM T67162 CP8RF4 46180256 Ki > 10000 nM T67162 CG8UK9 46180257 Ki > 10000 nM T67162 CO7SA6 46180258 Ki > 10000 nM T67162 CSY63N 46180259 Ki > 10000 nM T67162 C64TDV 46180261 Ki > 10000 nM T67162 CBM9O6 46180325 Ki > 10000 nM T67162 C1J3VH 46180327 Ki > 10000 nM T67162 CN3X9Q 46180328 Ki > 10000 nM T67162 C73KNC 46180331 Ki > 10000 nM T67162 CHN09F 46180394 Ki > 10000 nM T67162 CMS7T5 46180395 Ki > 10000 nM T67162 C62FUY 46180396 Ki > 10000 nM T67162 C10OKI 46180397 Ki > 10000 nM T67162 CM4R8A 46180398 Ki > 10000 nM T67162 CC7N8T 46180399 Ki > 10000 nM T67162 CLBT94 46190877 Ki = 5011.87 nM T67162 CSV1P2 46216855 Ki = 93 nM T67162 C5FQ4S 46224879 Ki = 34.67 nM T67162 COFU37 46225335 Ki > 10000 nM T67162 C9XTG3 46225336 Ki > 10000 nM T67162 C96LBQ 46225337 Ki > 10000 nM T67162 C6MC8Z 46225569 Ki > 3162.28 nM T67162 CS6Y9W 46225581 Ki = 39.81 nM T67162 C78DON 46225582 Ki = 398.11 nM T67162 CC8E3T 46225583 Ki = 79.43 nM T67162 CML42B 46225584 Ki = 794.33 nM T67162 CY7NM6 46227242 Ki = 2724 nM T67162 CR9S7B 46227243 Ki > 10000 nM T67162 C9A8FV 46227273 Ki = 7371 nM T67162 CL3KU2 46227284 Ki > 10000 nM T67162 CS4O6A 46227317 Ki = 320 nM T67162 CE1L6H 46227320 Ki > 10000 nM T67162 CSQ9D5 46227325 Ki > 10000 nM T67162 CX2Q1D 46228604 Ki = 38.02 nM T67162 CDI10H 46231541 Ki = 2000 nM T67162 CMR89A 46231588 Ki = 6000 nM T67162 CAW5U2 46231589 Ki = 2000 nM T67162 CBGM85 46231645 Ki = 552 nM T67162 C9KI4E 46231646 Ki = 5400 nM T67162 CYM51R 46231709 Ki = 1093 nM T67162 C8SFI5 46231768 Ki = 2100 nM T67162 C9BT2H 46231769 Ki = 2137 nM T67162 CD6T5Y 46231770 Ki = 1000 nM T67162 C3TIF9 46231771 Ki = 618 nM T67162 C0R6GH 46231772 Ki = 900 nM T67162 C1EW4S 46231782 Ki = 923 nM T67162 CF3NS8 46231783 Ki = 420 nM T67162 C6JM5T 46231784 Ki = 440 nM T67162 CFJP50 46231833 Ki = 500 nM T67162 CR9L3V 46231834 Ki = 1.3 nM T67162 C14XCV 46231835 Ki = 26 nM T67162 CD6IC3 46231845 Ki = 1693 nM T67162 C38WBY 46231846 Ki = 1371 nM T67162 C0A7GW 46231847 Ki = 1647 nM T67162 CVT82S 46231848 Ki = 1370 nM T67162 C9W1US 46231924 Ki = 483 nM T67162 CL7WX9 46231925 Ki = 217 nM T67162 CVG26Z 46231926 Ki = 69 nM T67162 CKJ09A 46231927 Ki = 124 nM T67162 CEMA94 46231992 Ki = 79 nM T67162 CLWO70 46231993 Ki = 223 nM T67162 C2BX8U 46231994 Ki = 584 nM T67162 C7FD2G 46231995 Ki = 618 nM T67162 C0IBN1 46232064 Ki = 1612 nM T67162 CM0PC8 46232065 Ki = 312 nM T67162 CYV52A 46232066 Ki = 550 nM T67162 CT8X1D 46232067 Ki = 12 nM T67162 C8XW1L 46232134 Ki = 89 nM T67162 CCL53R 46232135 Ki = 51 nM T67162 C9FV8B 46233097 Ki = 86 nM T67162 C24GSH 46233135 Ki = 41.4 nM T67162 C5TC2S 46830335 IC50 > 10000 nM T67162 C1K7FL 46830336 IC50 > 10000 nM T67162 C1N4KX 46842383 IC50 > 10000 nM T67162 C0WJ5L 46850462 Ki = 1700 nM T67162 CN3RH6 46850464 Ki = 250 nM T67162 CC62SX 46866711 IC50 > 10000 nM T67162 C03LTM 46869265 Ki = 230 nM T67162 CK8A1O 46880462 Ki > 10000 nM T67162 C9KDP4 46880463 Ki > 10000 nM T67162 CODR73 46880498 Ki > 10000 nM T67162 CHJ5Y6 46880566 Ki > 10000 nM T67162 CE9PG2 46880567 Ki > 10000 nM T67162 C01PGO 46880568 Ki > 10000 nM T67162 CS7L4X 46880569 Ki > 10000 nM T67162 C0PXY7 46880628 Ki > 10000 nM T67162 CD37LU 46880629 Ki > 10000 nM T67162 CUY89F 46880630 Ki > 10000 nM T67162 C4P6XS 46880631 Ki > 10000 nM T67162 CJ53KF 46880672 Ki > 10000 nM T67162 CYJC08 46880673 Ki > 10000 nM T67162 C1RI9O 46880674 Ki > 10000 nM T67162 CM2ZY5 46881408 EC50 = 10 nM T67162 C1R8WT 46881409 EC50 = 7.943 nM T67162 CT2VZ3 46881410 Ki = 630.96 nM T67162 CW62EC 46881411 EC50 = 125.89 nM T67162 CAHF16 46881412 EC50 = 125.89 nM T67162 CT9IF0 46881413 Ki = 630.96 nM T67162 C2MC4K 46881463 EC50 = 0.631 nM T67162 C27IES 46881464 Ki = 630.96 nM T67162 CP24SO 46881465 Ki = 630.96 nM T67162 C4Y9UE 46881466 Ki = 19.95 nM T67162 C9AJI3 46881467 EC50 = 501.19 nM T67162 C0EF4O 46882004 EC50 = 1 nM T67162 CR4CN8 46882005 EC50 = 2.512 nM T67162 CR9SO6 46882006 EC50 = 50.12 nM T67162 CJMC05 46882007 Ki = 0.631 nM T67162 CJYU26 46882008 Ki > 630.96 nM T67162 CAU9M8 46882009 EC50 = 10 nM T67162 CB34TO 46882049 Ki = 50.12 nM T67162 CDTA05 46882050 Ki = 39.81 nM T67162 CB13IH 46882051 Ki = 1.585 nM T67162 C0HM3E 46882052 EC50 = 0.631 nM T67162 CM93UE 46882053 EC50 = 0.7943 nM T67162 CDXI13 46882054 EC50 = 10 nM T67162 C4BH9E 46882458 Ki = 100 nM T67162 CF8IJ2 46882520 Ki = 398.11 nM T67162 CQN87I 46882521 Ki = 630.96 nM T67162 C56ULO 46882522 Ki = 630.96 nM T67162 CX72IN 46882583 Ki > 1000 nM T67162 CB8GE1 46884818 IC50 > 10000 nM T67162 C4MQ0A 46884856 IC50 > 10000 nM T67162 CCNT25 46884898 IC50 > 10000 nM T67162 C3MSG2 46885027 IC50 > 10000 nM T67162 CB7XI0 46885213 IC50 > 10000 nM T67162 CZR76I 46888925 Ki = 8.6 nM T67162 C4Q3SD 46888926 Ki = 8.6 nM T67162 CH9S8A 46888927 Ki = 8.3 nM T67162 C8T6WQ 46888928 Ki = 8 nM T67162 CJY47V 46888983 Ki = 9 nM T67162 CJ6IB7 46888984 Ki = 19 nM T67162 C18KHC 46888985 Ki = 2.5 nM T67162 CK40FT 46888986 Ki = 18 nM T67162 CTJ1P2 46889013 Ki = 9 nM T67162 COPQ75 46889014 Ki = 16 nM T67162 CAM45V 46889015 Ki = 6.3 nM T67162 CZ3FI5 46889016 Ki = 11 nM T67162 C4B6ZE 46889041 Ki = 7 nM T67162 CRW2I9 46893146 Ki = 6.9 nM T67162 C6BD5G 46905072 Ki = 170 nM T67162 CV9E5Y 46912547 Ki = 0.9 nM T67162 C34ILU 46912548 Ki = 0.9 nM T67162 CA75HK 46914485 Ki = 5122 nM T67162 C9D7UW 46914486 Ki = 5728 nM T67162 COB4R0 46914487 Ki = 2700 nM T67162 C4JZR8 46914620 Ki = 6005 nM T67162 C4JIP7 46914621 Ki = 4542 nM T67162 CZ5TS4 46914771 Ki = 4868 nM T67162 C1LY6Z 46914772 Ki > 10000 nM T67162 C3XE4P 46914773 Ki = 2281 nM T67162 C2E6UX 46914774 Ki > 10000 nM T67162 CT36AF 46914775 Ki = 2977 nM T67162 CW74CK 46914776 Ki > 10000 nM T67162 CLC27S 46914777 Ki > 10000 nM T67162 CAT12G 46914926 Ki = 2920 nM T67162 CE6SQ2 46914927 Ki > 10000 nM T67162 CGSN70 46917563 Ki = 4.1 nM T67162 CEH10Y 46917637 Ki = 8.8 nM T67162 CVQ01I 46929184 EC50 = 9 nM T67162 C7FX8L 46931072 Ki = 304 nM T67162 CKO76R 46931815 Ki = 398.11 nM T67162 CZDN92 46934426 Ki = 254 nM T67162 C4VG2E 46934427 Ki = 99 nM T67162 CUTX67 46934428 IC50 > 10000 nM T67162 C6J4TV 46946859 Ki = 7.39 nM T67162 C3XFG4 47029237 Ki > 10000 nM T67162 CY28OS 47556338 Ki = 5848 nM T67162 CYWX19 49780808 Ki = 251.19 nM T67162 C9RI3L 49780809 Ki = 501.19 nM T67162 C39KWP 49781039 Ki > 3162.28 nM T67162 C9O2RB 49781040 Ki = 199.53 nM T67162 C95ZVI 49781232 Ki = 0.44 nM T67162 C7T9AD 49781234 Ki = 0.86 nM T67162 CAE6P4 49781235 Ki = 1.6 nM T67162 C5GL9U 49781236 Ki = 2.3 nM T67162 C7T3KS 49781255 Ki = 125.89 nM T67162 C2RE4X 49781447 Ki = 5.9 nM T67162 CPH42B 49781448 Ki = 2.9 nM T67162 CIOK26 49781449 Ki = 1.9 nM T67162 CW41PI 49781450 Ki = 0.62 nM T67162 CFM61E 49781451 Ki = 1.1 nM T67162 CJN1B3 49781452 Ki = 0.73 nM T67162 C0BFH7 49781453 Ki = 1.8 nM T67162 CYL65E 49781476 Ki = 398.11 nM T67162 CFQN89 49781477 Ki > 3162.28 nM T67162 CL82ES 49781478 Ki > 3162.28 nM T67162 C5NBV9 49781676 Ki = 1.6 nM T67162 C7FOU5 49781677 Ki = 3.4 nM T67162 CT1IQ8 49781678 Ki = 6.3 nM T67162 CI43JH 49781679 Ki = 2 nM T67162 C3S4MB 49781680 Ki = 4.6 nM T67162 CB14EV 49781681 Ki = 4.9 nM T67162 CU8V4W 49781890 Ki = 0.35 nM T67162 CAY72O 49781891 Ki = 1.9 nM T67162 C9TE7L 49781892 Ki = 7.1 nM T67162 CQ1F6E 49781893 Ki = 12 nM T67162 CDJ9E3 49781894 Ki = 6.1 nM T67162 CESC01 49782398 Ki = 3.6 nM T67162 C8BWU1 49782600 Ki = 3.4 nM T67162 C6I0NJ 49782601 Ki = 13 nM T67162 C20CVH 49782602 Ki = 140 nM T67162 CY4FW1 49782603 Ki = 15 nM T67162 CXJ59F 49782604 Ki = 46 nM T67162 CPFY62 49782791 Ki = 27 nM T67162 CKGU71 49782792 Ki = 3.3 nM T67162 CNE84I 49782794 Ki = 31 nM T67162 CD9ZH7 49782836 Ki = 19 nM T67162 CL1J4C 49782837 Ki = 440 nM T67162 CB53QP 49782841 Ki = 83 nM T67162 CS09QO 49782998 Ki = 4.5 nM T67162 CENR09 49783039 Ki = 65 nM T67162 CZ5G9J 49783040 Ki = 17 nM T67162 C98JVY 49783041 Ki = 32 nM T67162 CRML65 49783042 Ki = 86 nM T67162 COM8D5 49798797 Ki = 61 nM T67162 C9ZYH8 49798799 Ki = 254 nM T67162 C4TXW8 49798812 Ki = 14.3 nM T67162 C9KOV8 49798833 Ki = 46.8 nM T67162 C6LP9T 49798835 Ki = 6.6 nM T67162 C6RE1F 49798837 Ki = 2.4 nM T67162 CMQ23B 49798839 Ki = 13.6 nM T67162 C2WZ9Y 49798853 Ki = 37.8 nM T67162 CU34RI 49798855 Ki = 7.1 nM T67162 CM86YK 49798857 Ki = 8 nM T67162 CTDN46 49798874 Ki = 2 nM T67162 CO4K6F 49798877 Ki = 4.2 nM T67162 C69EKV 49798878 Ki = 4.2 nM T67162 CWQ9Y1 49798879 Ki = 2.5 nM T67162 CV1S3H 49799687 Ki = 3.8 nM T67162 CBR67S 49799691 Ki = 1396 nM T67162 C5A6TG 49799693 Ki = 13.8 nM T67162 CZ8A2G 49799695 Ki = 23.3 nM T67162 CCV35T 49799709 Ki = 27.7 nM T67162 CLY02B 49799713 Ki = 12.5 nM T67162 CDTS15 49799715 Ki = 212 nM T67162 CDAB96 49836026 Ki = 501.19 nM T67162 CR40BA 49836386 IC50 > 30000 nM T67162 C0M5XC 49836496 IC50 > 30000 nM T67162 C4R2YS 49850567 Ki = 199.53 nM T67162 C07JTU 49850570 Ki = 316.23 nM T67162 CK68QR 49850672 Ki = 199.53 nM T67162 CN5XR1 49850772 Ki = 398.11 nM T67162 CR4EZ0 49850870 Ki = 398.11 nM T67162 C5K4EC 49850872 Ki = 398.11 nM T67162 C8AW0R 49850874 Ki = 398.11 nM T67162 C6OQV2 49862237 Ki > 1000 nM T67162 CDHY90 49864027 Ki > 10000 nM T67162 C9KIU1 49864289 IC50 > 10000 nM T67162 CHO9C0 49864292 IC50 > 10000 nM T67162 C8TB6G 49864336 Ki = 46.5 nM T67162 C5N8ML 49864359 Ki = 438 nM T67162 C15NIO 49864360 Ki = 121 nM T67162 C90MTG 49864602 IC50 > 10000 nM T67162 C5BCS4 49864722 IC50 > 10000 nM T67162 CKZO79 49864723 IC50 > 10000 nM T67162 C74LZS 49864724 IC50 > 10000 nM T67162 CKWA93 49865589 Ki = 501.19 nM T67162 C8J5PI 49865599 Ki = 0.8 nM T67162 CP63AX 49865600 Ki = 0.4 nM T67162 CA1IY0 49865601 Ki = 17 nM T67162 CXWL20 49865623 Ki = 501.19 nM T67162 CC5KD7 49865639 Ki = 11 nM T67162 C1B5RD 49865640 Ki = 32 nM T67162 C51PJT 49865641 Ki = 12 nM T67162 C3KF6B 49865668 Ki = 1 nM T67162 C2RY0J 50878551 Ki > 10000 nM T67162 C1W6TV 50898777 Ki > 10000 nM T67162 CXMZ73 50898778 Ki > 10000 nM T67162 CX48AD 51002362 Ki = 1812 nM T67162 C8TA1J 51003550 IC50 = 136 nM T67162 CQ1UJ7 51003551 IC50 > 10000 nM T67162 CGMI37 51003586 IC50 > 1000 nM T67162 CE4KP1 51050257 Ki > 10000 nM T67162 CIJT81 51111982 Ki = 1821 nM T67162 C2HGK8 51122451 Ki > 1000 nM T67162 CMYT24 51353673 Ki = 20.9 nM T67162 C5W4PN 51353674 Ki = 13.2 nM T67162 C0UBA8 51353675 Ki = 57.6 nM T67162 CU3C4O 51353676 Ki = 15.1 nM T67162 CB3A9S 51353677 Ki = 21.4 nM T67162 C1LHZ4 51353678 Ki = 15.1 nM T67162 CIO10J 51353988 Ki = 14.2 nM T67162 CWFU41 51353989 Ki = 0.17 nM T67162 CA01KY 51353990 Ki = 31.7 nM T67162 CA8E9Q 51353991 Ki = 35.2 nM T67162 CW8LE6 51353992 Ki = 17.7 nM T67162 CL8WR0 51354273 Ki = 37.9 nM T67162 CW03GI 51354274 Ki = 64.8 nM T67162 C2DG1Z 51354275 Ki = 70.5 nM T67162 CT8MC6 51354277 Ki = 27.1 nM T67162 CEL30Q 51354279 Ki = 131 nM T67162 CU9B6W 51354566 Ki = 55.3 nM T67162 COD5H3 51354851 Ki = 52 nM T67162 CPN8T3 51354853 Ki = 59.2 nM T67162 C7Q2MW 51355139 Ki = 17.8 nM T67162 CMYZ04 51355143 Ki = 13.4 nM T67162 CI5Q4B 51356569 EC50 = 951 nM T67162 C42GMN 52937680 Ki = 240 nM T67162 C96LHK 52937776 Ki = 77 nM T67162 C30RKG 52937777 Ki = 43 nM T67162 C78FZD 52937871 Ki = 4700 nM T67162 C1S9VT 52937875 Ki = 49 nM T67162 CFK1D4 52937876 EC50 = 0.51 nM T67162 CIWA18 52938727 Ki = 7384 nM T67162 C6XY8V 52938728 Ki = 661 nM T67162 C9C0NB 52940734 Ki = 9.44 nM T67162 CJ19FP 52940753 Ki = 2511.89 nM T67162 CCDZ51 52940788 Ki = 199.53 nM T67162 C2RW5A 52940961 Ki = 398.11 nM T67162 CS5I2W 52940985 Ki = 190 nM T67162 CCK37R 52941006 EC50 = 52.6 nM T67162 CQP43J 52941038 IC50 = 57.54 nM T67162 C1NJ5B 52941039 IC50 = 25.7 nM T67162 C7VRX0 52941040 IC50 = 7.762 nM T67162 CBS38E 52941042 IC50 = 7.079 nM T67162 C1ZGF5 52941075 IC50 = 1.096 nM T67162 CHOA42 52941076 IC50 = 1.288 nM T67162 C9IJ4D 52941078 IC50 = 19.95 nM T67162 C0UXM7 52941358 Ki = 35.2 nM T67162 CTM81E 52941423 Ki = 3.03 nM T67162 C8FZL4 52941427 Ki = 316.23 nM T67162 CCL40E 52941643 IC50 = 204.17 nM T67162 CM4XO6 52941718 Ki = 22 nM T67162 C8E1MB 52941809 Ki = 24 nM T67162 C0BK7I 52942259 IC50 = 2.884 nM T67162 C6H5BR 52942266 IC50 = 141.25 nM T67162 CEZM65 52942303 IC50 = 0.2884 nM T67162 C0XBE8 52942307 IC50 = 1.778 nM T67162 CHN17C 52942381 Ki = 35 nM T67162 CRI12K 52942395 Ki = 120 nM T67162 CE6R7D 52942615 Ki = 6.81 nM T67162 CX2E5H 52942854 Ki = 58 nM T67162 CU8WA5 52942916 Ki = 33.8 nM T67162 C4PQ7Z 52942934 IC50 = 65 nM T67162 CS52JH 52943464 IC50 = 0.912 nM T67162 CX52QY 52943468 IC50 = 10.96 nM T67162 C09RJS 52943802 Ki = 260 nM T67162 CT78RV 52944077 IC50 = 5.495 nM T67162 C2IA0W 52944078 IC50 = 16.98 nM T67162 CBU2Z6 52944379 Ki = 21.8 nM T67162 C5HQ2F 52944651 IC50 = 16.98 nM T67162 CCT4Q9 52944652 IC50 = 2.291 nM T67162 CG7WJ9 52944653 IC50 = 67.61 nM T67162 CL58OI 52944655 IC50 = 70.79 nM T67162 CT13RE 52944656 IC50 = 10.96 nM T67162 CYH67R 52944657 IC50 = 3019.95 nM T67162 C49AOG 52944701 IC50 = 186.21 nM T67162 CQJ7C0 52945023 Ki > 3162.28 nM T67162 C59ASG 52945060 Ki = 13.6 nM T67162 CT51OC 52945819 Ki = 13 nM T67162 C4SH8M 52945840 Ki = 0.812 nM T67162 C0J6VC 52945902 IC50 = 5.623 nM T67162 C8NPC7 52945904 IC50 = 64.57 nM T67162 CA9G6V 52945905 IC50 = 25.7 nM T67162 CQ1I6V 52945907 IC50 = 3.236 nM T67162 CRH43M 52946023 Ki = 3.1 nM T67162 COZ9J3 52946432 Ki = 100 nM T67162 C19ZKQ 52946556 Ki = 17.5 nM T67162 CRIV53 52946792 Ki = 1.7 nM T67162 C4S8JC 52946835 Ki = 2.46 nM T67162 CI31VP 52947113 IC50 = 316.23 nM T67162 C2AK9B 52947114 IC50 = 4.169 nM T67162 CF7Q0X 52947123 IC50 = 32.36 nM T67162 C8OSX3 52947124 IC50 = 56.23 nM T67162 CV0UI1 52947127 IC50 = 109.65 nM T67162 CI0K9N 52947128 IC50 = 123.03 nM T67162 CS3OD1 52947342 Ki = 9.01 nM T67162 CCOQ59 52947343 Ki = 9.86 nM T67162 C6YB2T 52947380 Ki = 51.6 nM T67162 CI5V3X 52947507 Ki = 3162.28 nM T67162 C6ZSQ8 52947516 Ki = 316.23 nM T67162 CN32PV 52947694 Ki = 100 nM T67162 CUV0G4 52947756 Ki = 17 nM T67162 CD17LV 52948101 Ki = 16.6 nM T67162 C7IR4Q 52948256 Ki = 3.81 nM T67162 CT27HL 52948318 IC50 = 363.08 nM T67162 CBLE49 52948319 IC50 = 38.9 nM T67162 C73RXF 52948320 IC50 = 12.02 nM T67162 C1M9BF 52948326 IC50 = 7.943 nM T67162 CJ6OP5 52948620 Ki = 5.91 nM T67162 CZ01DH 52948653 Ki = 398.11 nM T67162 C9OSI0 52949300 Ki = 199.53 nM T67162 CLOB90 52949351 Ki = 2.34 nM T67162 CZ3C9K 52949578 IC50 = 1.514 nM T67162 C8BWP7 52949580 IC50 = 1.698 nM T67162 CHF68S 52949582 IC50 = 19.05 nM T67162 C9WLF6 52949583 IC50 = 5.012 nM T67162 C3ZC2U 52949614 IC50 = 3.02 nM T67162 C0RUM1 52949810 Ki = 9.31 nM T67162 CS6O4B 52949885 Ki = 13.1 nM T67162 CILY85 52950060 Ki = 10.6 nM T67162 C45SNB 52950130 IC50 = 10.96 nM T67162 CPVM58 52950169 Ki = 24.5 nM T67162 C4IV2J 53248158 Ki = 390 nM T67162 C03JEZ 53248159 Ki = 378 nM T67162 C2G0ZY 53248208 Ki = 329 nM T67162 C2UKM3 53248209 Ki = 960 nM T67162 C8KW9J 53248210 Ki = 274 nM T67162 C87SLP 53248211 Ki = 279 nM T67162 CVD7E5 53248212 Ki = 421 nM T67162 CX6KG9 53248213 Ki = 526 nM T67162 C63MQD 53248256 Ki = 2890 nM T67162 CG2O7F 53248257 Ki = 4260 nM T67162 CRK87G 53248258 Ki = 241 nM T67162 C73WQX 53248259 Ki = 472 nM T67162 CKOV84 53248260 Ki = 302 nM T67162 C09IXA 53248261 Ki = 230 nM T67162 C5K7NT 53248298 Ki = 195 nM T67162 C28DOY 53248299 Ki = 84 nM T67162 CIM15A 53248300 Ki = 15.6 nM T67162 C0LS5Y 53248345 Ki = 196 nM T67162 CSU1D5 53248346 Ki = 269 nM T67162 CBS3U2 53248347 Ki = 119 nM T67162 C85RJF 53248348 Ki = 313 nM T67162 CF3AO9 53248349 Ki = 2090 nM T67162 CSF8M1 53248393 Ki = 5270 nM T67162 C6P5WJ 53248394 Ki = 869 nM T67162 CN4SY6 53248395 Ki = 2060 nM T67162 CC78FG 53248673 Ki = 0.26 nM T67162 CL3WJ1 53248675 Ki = 0.14 nM T67162 CG6T2N 53248677 Ki = 0.07 nM T67162 C8DSO1 53304086 Ki = 53.7 nM T67162 C5C8ZN 53317208 Ki = 206 nM T67162 CSM53O 53317282 Ki = 616 nM T67162 CA31DT 53318564 Ki = 399 nM T67162 CU4CR9 53318565 Ki = 174 nM T67162 C61DNP 53320009 IC50 > 10000 nM T67162 C9ZDR5 53320010 IC50 > 10000 nM T67162 C5DL8F 53321194 Ki = 141 nM T67162 C3M6UO 53322449 Ki = 1203 nM T67162 CHU18S 53322522 Ki = 293 nM T67162 CQLK01 53322638 IC50 = 1784 nM T67162 C3B4SQ 53323859 Ki = 600 nM T67162 C32YWL 53324045 Ki = 38 nM T67162 C35GJZ 53325137 Ki = 88 nM T67162 CB6RV7 53325138 Ki = 770 nM T67162 CRQF15 53325242 Ki = 194 nM T67162 C0UC1W 53326601 Ki = 34.4 nM T67162 CV2I6F 53327181 Ki = 660 nM T67162 C9KH8Y 53327217 Ki = 140 nM T67162 C34YFD 53327218 Ki = 570 nM T67162 CY4HB1 53327219 Ki = 109.65 nM T67162 C3LOV2 53327220 Ki = 309.03 nM T67162 CB96WM 53327221 Ki = 97.72 nM T67162 CI89KJ 53327222 Ki = 23.99 nM T67162 C5FYM1 53327260 Ki = 128.82 nM T67162 CPN87B 53327261 Ki = 199.53 nM T67162 C3PO5L 53327262 Ki = 0.2291 nM T67162 CQR72D 53327263 Ki = 120.23 nM T67162 CS5Z7X 53327908 Ki = 7.1 nM T67162 C5TVA7 53359024 Ki > 10000 nM T67162 CLZ09P 53359025 Ki = 1724 nM T67162 CPQ1E2 53361301 Ki = 22 nM T67162 CABK98 53361302 Ki = 12 nM T67162 CBF2P3 53362655 Ki = 871 nM T67162 C9MK6L 53362715 Ki = 2005 nM T67162 C47KPJ 53362716 Ki = 2200 nM T67162 CLP09I 53362717 Ki = 851 nM T67162 C7PA6D 53362719 Ki = 352 nM T67162 C8GC1B 53362840 Ki = 2800 nM T67162 CU7W2I 53362841 Ki = 4300 nM T67162 CK0M7F 53363109 Ki = 63 nM T67162 CG24FV 53363110 Ki = 52 nM T67162 CD8C0B 53363111 Ki = 69 nM T67162 C28MPE 53363199 Ki = 68 nM T67162 CN3C4E 53363200 Ki = 16 nM T67162 CYW7M4 53363201 Ki = 7.3 nM T67162 C6EU7I 53363202 Ki = 17 nM T67162 CMI25H 53364083 Ki = 32 nM T67162 C1UWI5 53364153 Ki = 16 nM T67162 C78PUJ 53364154 Ki = 17 nM T67162 CRB76A 53364155 Ki = 8.2 nM T67162 CZV06L 53364225 Ki = 3.3 nM T67162 CQ7PX0 53364226 Ki = 2.8 nM T67162 CCA02T 53364227 Ki = 4.8 nM T67162 CU4B6N 53370045 Ki = 2130 nM T67162 CEIG81 53391632 Ki = 1350 nM T67162 CQ3M2A 53391731 Ki = 1489 nM T67162 CMOZ61 53475319 Ki = 21 nM T67162 CQG92V 53483975 Ki > 10000 nM T67162 CWH50X 53499206 Ki > 10000 nM T67162 C7HP2L 53524618 Ki > 10000 nM T67162 C9PQ6Y 53550713 Ki > 10000 nM T67162 CR07QE 54186017 Ki > 1600 nM T67162 C0JC2O 54325398 Ki = 25.12 nM T67162 CX7H3P 54325399 Ki = 100 nM T67162 CNG7U0 54434812 Ki = 34 nM T67162 CV2G4S 54437013 Ki = 1584.89 nM T67162 C5JL8O 54437014 Ki = 501.19 nM T67162 CL5QO2 54493650 Ki = 501.19 nM T67162 CCM43W 54580387 Ki = 162 nM T67162 CKND43 54580905 Ki = 15 nM T67162 CF6G4L 54580906 Ki = 4.8 nM T67162 CHNI24 54581963 Ki = 0.93 nM T67162 CM5TK0 54581964 Ki = 2.1 nM T67162 C8AT1S 54583897 Ki = 9.2 nM T67162 CW9Z2J 54583898 Ki = 8.8 nM T67162 CN6O2E 54584336 Ki = 69.9 nM T67162 C8V6BJ 54584468 Ki = 914 nM T67162 CY9QZ8 54584591 Ki = 38 nM T67162 CIMS79 54585306 Ki = 64.7 nM T67162 CU3M5C 54585745 Ki > 10000 nM T67162 CL23NI 54585810 Ki = 52 nM T67162 CW1I5B 54585811 Ki = 22 nM T67162 CTQ08M 54586179 Ki = 3 nM T67162 C3QJP1 54735210 Ki = 25.5 nM T67162 CL5I1R 54753271 Ki = 870 nM T67162 COZ82F 55479093 Ki = 84 nM T67162 CY27RS 56360144 IC50 > 100000 nM T67162 CFV6N1 56361664 IC50 = 691 nM T67162 CF59RX 56361674 EC50 > 50000 nM T67162 CQ3AR0 56589560 Ki = 85.3 nM T67162 C4XGR3 56589561 Ki = 2923 nM T67162 C9PHZ3 56594402 Ki > 10000 nM T67162 C82IVX 56594533 Ki > 10000 nM T67162 CT4J5C 56594534 Ki = 268 nM T67162 CW89BT 56595402 Ki > 1000 nM T67162 C4C3XQ 56595529 Ki > 1000 nM T67162 CA54LD 56597090 Ki = 42 nM T67162 C1DB3K 56597091 Ki = 66 nM T67162 CSQ54O 56597092 Ki = 18 nM T67162 C57NES 56597095 Ki = 15 nM T67162 C38MNW 56597225 Ki = 17 nM T67162 CG0K6E 56597637 Ki = 3.236 nM T67162 CR96VY 56597939 Ki = 104 nM T67162 CLH68F 56598070 Ki = 18 nM T67162 CJ29WT 56598071 Ki = 20 nM T67162 C0M4HB 56599143 Ki = 30 nM T67162 C7SO9N 56599144 Ki = 11 nM T67162 C7MRL8 56599145 EC50 = 4 nM T67162 CV4FI7 56599146 Ki = 145 nM T67162 CF07US 56599147 EC50 = 199 nM T67162 CJ57IF 56658006 Ki = 309 nM T67162 CTWV58 56658008 Ki = 7.4 nM T67162 CY7L0C 56658155 Ki = 1648 nM T67162 CFD2M9 56658156 Ki = 5866 nM T67162 CD51XT 56658157 Ki = 89 nM T67162 C8RWM0 56661666 Ki = 484 nM T67162 CU2C6F 56663238 IC50 > 2511.89 nM T67162 C1CJ8P 56664948 Ki = 145 nM T67162 C26RNX 56664950 Ki = 25.3 nM T67162 CRPA72 56664952 Ki = 7.3 nM T67162 C0CS2Z 56670092 IC50 = 2511.89 nM T67162 C7D6LT 56670158 IC50 > 3162.28 nM T67162 CXC4G1 56673609 IC50 = 1995.26 nM T67162 CRSF93 56673674 IC50 = 794.33 nM T67162 CW7F5G 56675269 Ki = 102 nM T67162 CY6D5E 56675412 Ki = 1025 nM T67162 C4B2UC 56675413 Ki = 432 nM T67162 CC2B8F 56678599 Ki = 2604 nM T67162 CEV53O 56678761 Ki = 556 nM T67162 C28ECA 56681925 Ki = 611 nM T67162 CLX25U 56681927 Ki = 4.6 nM T67162 C8H1LP 56682068 Ki = 5791 nM T67162 CK9SG4 56781741 Ki = 5596 nM T67162 CY2S8M 56820088 Ki = 3231 nM T67162 CFE60O 56833378 Ki = 16 nM T67162 C04VKH 56833379 Ki = 110 nM T67162 CAS80D 56833463 Ki = 12 nM T67162 CUXP15 56833464 Ki = 17 nM T67162 C6DEW7 56837419 Ki = 14 nM T67162 CZ1WY0 56837634 Ki = 25 nM T67162 CKJ2U0 56837635 Ki = 16 nM T67162 CZP6E4 56837636 Ki = 6.4 nM T67162 CXJ7R9 56926585 Ki = 16000 nM T67162 CH1S9B 56926586 Ki = 6100 nM T67162 CJ42HS 56926587 Ki = 29000 nM T67162 C1ZG7A 56933434 Ki = 16 nM T67162 C7G5PJ 56941366 EC50 = 15.9 nM T67162 CO0N2W 56943599 Ki = 51 nM T67162 C3DF5Z 56943600 Ki = 1 nM T67162 C19BDH 56943695 Ki = 8 nM T67162 CS7K3T 56943891 Ki = 27 nM T67162 CZ4L3S 56944082 Ki = 77 nM T67162 C5NI3K 56944086 Ki = 5.3 nM T67162 C37BYO 56944186 Ki = 54 nM T67162 C9UOZ6 56944189 Ki = 100 nM T67162 CH7V9J 56944190 Ki = 15 nM T67162 CE49MC 56944191 Ki = 26 nM T67162 CX2RP5 56944287 Ki = 64 nM T67162 CB0P9N 56944383 Ki = 1.8 nM T67162 CEQ7I3 56944384 Ki = 1.2 nM T67162 CHWI01 56944473 Ki = 25 nM T67162 C6Y4ZQ 56944564 Ki = 0.9 nM T67162 C3B0MZ 56944565 Ki = 8.7 nM T67162 CI4KW0 56944664 Ki = 44 nM T67162 C39YHD 56944665 Ki = 3 nM T67162 C1W3GL 56944666 Ki = 1.1 nM T67162 C7J4UT 56944667 Ki = 17 nM T67162 CZT80U 56944668 Ki = 1 nM T67162 CTW2F5 56944763 Ki = 5.2 nM T67162 C50WEX 56944764 Ki = 20 nM T67162 CX0ZW2 56944859 Ki = 9.1 nM T67162 C1ST9U 56944860 Ki = 2.3 nM T67162 CQKL90 56944861 Ki = 2.6 nM T67162 CS5J6Y 56944862 Ki = 4.5 nM T67162 CFLB40 56944863 Ki = 1 nM T67162 C53OTR 56944864 Ki = 2.5 nM T67162 C5T3RI 56944951 Ki = 2.8 nM T67162 CR6H7U 56944952 Ki = 3.5 nM T67162 C1Y2RP 56944953 Ki = 2.7 nM T67162 C1BH7I 56944954 Ki = 2.6 nM T67162 CTK9I8 56944955 Ki = 37 nM T67162 CCF1A5 56944956 Ki = 2.4 nM T67162 C2YVT8 56945042 Ki = 11 nM T67162 CNI2G3 56945043 Ki = 23 nM T67162 CF9V3Q 56945045 Ki = 49 nM T67162 CE4S5M 56945046 Ki = 6 nM T67162 C1TC7Q 56963799 Ki > 10000 nM T67162 CPT03G 57300602 Ki = 109 nM T67162 C8IC7Y 57325596 IC50 > 10000 nM T67162 C0V6CZ 57325597 IC50 > 10000 nM T67162 C7BLT2 57325598 IC50 > 10000 nM T67162 CLIV06 57325768 IC50 = 1617 nM T67162 CO1L7G 57326593 IC50 = 2398.83 nM T67162 CS6BD7 57326688 IC50 = 776 nM T67162 CG54VA 57326689 IC50 = 8912.51 nM T67162 CN5EY4 57326691 IC50 = 1778.28 nM T67162 C9B2KZ 57326789 IC50 > 10000 nM T67162 C68UZW 57326790 IC50 > 10000 nM T67162 CPWU35 57326791 IC50 > 10000 nM T67162 CQ79JC 57326889 IC50 > 10000 nM T67162 CZY02A 57326890 IC50 > 10000 nM T67162 CM8E2L 57326891 IC50 = 2078 nM T67162 CB65TD 57326982 IC50 = 2440 nM T67162 C1BF4R 57326983 IC50 > 10000 nM T67162 CCU82V 57326984 IC50 > 10000 nM T67162 CD9I4N 57334553 IC50 = 26.3 nM T67162 CDZU04 57335757 EC50 = 14000 nM T67162 C6H9UV 57345617 Ki = 33 nM T67162 CZU6L2 57345618 Ki = 172 nM T67162 CK9G8H 57345619 Ki = 139 nM T67162 CU2M7Q 57345620 Ki = 180 nM T67162 C6QAE5 57383397 Ki = 530 nM T67162 C0KR7X 57383401 Ki = 210 nM T67162 C6NCE0 57383405 Ki = 240 nM T67162 CQO45V 57383408 Ki > 50000 nM T67162 C7XJ1A 57383414 Ki = 23 nM T67162 CMW19O 57383430 Ki = 90 nM T67162 CL8N9J 57383431 Ki = 190 nM T67162 CT5O6F 57383434 Ki = 290 nM T67162 C7LQV0 57383436 Ki = 310 nM T67162 C0QM2U 57390115 Ki = 44 nM T67162 CZ12PI 57390116 Ki = 1.8 nM T67162 CRG2X7 57390117 Ki = 320 nM T67162 CR9L2W 57390118 Ki = 11 nM T67162 C26DAH 57390119 Ki = 32 nM T67162 C6S0IE 57390695 Ki = 1983 nM T67162 C5OJP0 57391102 IC50 > 30000 nM T67162 CV08WY 57391216 Ki = 424 nM T67162 CD75YK 57391306 Ki = 998 nM T67162 C07PMA 57391307 Ki = 390 nM T67162 C53OMP 57391554 IC50 = 794.33 nM T67162 C0T9UH 57391895 Ki = 19 nM T67162 CPN87T 57391896 Ki = 20 nM T67162 C64AWK 57391897 Ki = 6.4 nM T67162 CWT20M 57393083 Ki = 269 nM T67162 C1M4PZ 57393627 Ki = 66 nM T67162 C7E4BW 57393628 Ki = 0.59 nM T67162 CGWK23 57393634 Ki = 270 nM T67162 CADH19 57394285 Ki = 751.1 nM T67162 C0WA3H 57394810 Ki = 185 nM T67162 CMNZ07 57394992 IC50 = 500 nM T67162 CYZD14 57395043 IC50 > 7943.28 nM T67162 C39YHG 57395340 Ki = 83 nM T67162 C35RST 57395341 Ki = 32 nM T67162 CD4A3P 57396484 Ki = 636 nM T67162 C4EXS6 57396571 Ki = 446.68 nM T67162 C3GW6L 57398351 Ki = 41 nM T67162 CO50ZB 57398352 Ki = 4753 nM T67162 C2CEB9 57398562 IC50 = 2511.89 nM T67162 C5YZM2 57398875 Ki = 3.9 nM T67162 CJ41PW 57399432 Ki = 258.7 nM T67162 CO3B4P 57399494 Ki = 1021 nM T67162 C1NGZ7 57400229 IC50 = 398.11 nM T67162 CI9XS8 57400556 Ki = 3 nM T67162 C20IPH 57400557 Ki = 12 nM T67162 CU0C3D 57400562 Ki = 9700 nM T67162 C3TYE1 57401435 IC50 > 10000 nM T67162 CM7EN2 57401436 IC50 = 1995.26 nM T67162 CZX05B 57401706 Ki = 183 nM T67162 CYN38R 57401819 Ki = 284 nM T67162 CO0XD2 57401820 Ki = 211 nM T67162 CO04CI 57402365 Ki = 140 nM T67162 C27OEI 57402366 Ki = 4.6 nM T67162 CFJ27E 57402787 Ki = 2.7 nM T67162 CX0B5M 57403525 Ki = 5.37 nM T67162 CWBG94 57403981 Ki = 44 nM T67162 CQ5A8S 57420188 EC50 = 0.389 nM T67162 CQB6F9 57456630 Ki > 1000 nM T67162 C9PLU4 57527911 Ki = 13400 nM T67162 CH3T2M 57587922 Ki = 1740 nM T67162 C0M5PN 57873490 Ki > 1000 nM T67162 CH1BN8 57873491 Ki > 1000 nM T67162 CI5UO1 57873492 Ki > 1000 nM T67162 C2D9HA 57873499 Ki = 1 nM T67162 C81MLX 57873504 Ki > 1000 nM T67162 C7L9IE 57873508 Ki > 1000 nM T67162 CZRL39 57873513 Ki > 1000 nM T67162 C98WTS 57873515 Ki > 1000 nM T67162 C6BHT3 57873518 Ki > 1000 nM T67162 CPX17D 57873520 Ki = 58 nM T67162 C54ROE 57873522 Ki > 1000 nM T67162 CM7PI1 57873525 Ki > 1000 nM T67162 CMUR21 57873527 Ki = 3412 nM T67162 CO5Y9Q 57873531 Ki = 85 nM T67162 CCX12B 58358826 Ki = 3.4 nM T67162 CJ0AR3 58765508 EC50 = 0.6 nM T67162 C2AY1P 60148494 EC50 = 114 nM T67162 CIFJ86 60148495 EC50 = 70.7 nM T67162 CHJL24 60148496 EC50 = 86.4 nM T67162 CEY2I7 60148497 EC50 = 2.96 nM T67162 C4MV2N 60149678 Ki > 100000 nM T67162 CYSV60 60165411 Ki = 505 nM T67162 CB9GC6 60165412 Ki = 198 nM T67162 CI5PM3 60165413 Ki = 642 nM T67162 C2Q5VD 60165416 Ki = 219 nM T67162 C9JL3F 60165418 Ki = 26.5 nM T67162 C31PEN 60165535 Ki = 30.8 nM T67162 CP60YF 60165537 Ki = 990 nM T67162 CP1DR8 60165539 Ki = 8355 nM T67162 C85OTH 60165541 Ki = 530 nM T67162 CJO91V 60165543 Ki = 1522 nM T67162 CJDC53 60165545 Ki = 2931 nM T67162 C3K5JN 60165681 Ki = 4793 nM T67162 C9Q7MR 60165801 EC50 = 114 nM T67162 C5RUP6 60167166 Ki = 2321 nM T67162 CRH49P 60167309 Ki = 199.53 nM T67162 CX0NY3 60167310 Ki > 10000 nM T67162 COHK72 60167451 Ki = 217 nM T67162 C30SVG 60167452 Ki = 25 nM T67162 CI30FT 60204111 Ki = 219 nM T67162 CWSA08 60204112 Ki > 1000 nM T67162 CXI15A 60481587 IC50 > 50000 nM T67162 C02TAQ 62705172 Ki = 2200 nM T67162 CV0X4K 62705173 Ki = 1100 nM T67162 CWL9J4 62705175 Ki = 600 nM T67162 CQ5LS1 62705176 Ki = 16 nM T67162 CK2DG6 62705177 Ki = 55 nM T67162 C59QUB 62705330 Ki = 1250 nM T67162 CANL67 62705331 Ki > 9500 nM T67162 CW19CI 62705332 Ki = 1350 nM T67162 CK2WS1 62705333 Ki = 650 nM T67162 C1SNE7 62705334 Ki = 60 nM T67162 C2O6FQ 62705335 Ki = 6.5 nM T67162 CTM29C 62705504 Ki = 90 nM T67162 CZHO61 62705505 Ki = 95 nM T67162 CT41VY 62705506 Ki = 41 nM T67162 CP9HO0 62705507 Ki = 14 nM T67162 CSHR51 62705508 Ki = 2.5 nM T67162 CVPW40 62705509 Ki = 15 nM T67162 CM0Z3B 62707610 Ki = 9.5 nM T67162 CE5UK6 66559506 Ki = 113 nM T67162 CJ6B9Y 66559507 Ki = 108 nM T67162 CBS92F 66559587 Ki = 5.7 nM T67162 CG4VT2 66559588 EC50 = 2.5 nM T67162 C9AC7T 66559777 EC50 = 2.5 nM T67162 CI06XW 66559778 EC50 = 10 nM T67162 CJ0BI3 66559782 EC50 = 2 nM T67162 CLXS32 66561333 Ki = 3.6 nM T67162 CM24PO 66561413 Ki = 3575 nM T67162 CW36YC 66561968 Ki > 10000 nM T67162 CG5BP2 66574145 Ki = 148 nM T67162 C6AUO2 66800823 Ki = 8.3 nM T67162 C34ACQ 66800909 Ki = 27 nM T67162 CGT9E6 66800910 Ki > 1000 nM T67162 C0QY7D 66800916 Ki = 44 nM T67162 CM58FG 66800926 Ki > 10000 nM T67162 CQ43WD 66800934 Ki = 48 nM T67162 CK0I5J 66800939 Ki = 2.2 nM T67162 C0X2SF 66800942 Ki = 43 nM T67162 CN30YT 66800947 Ki = 10 nM T67162 CZ3MR6 66800959 Ki = 20 nM T67162 C92CMO 66800965 Ki = 1.8 nM T67162 CFPK92 66800991 Ki = 26 nM T67162 C13GMO 66801000 Ki = 48 nM T67162 CZ1TF9 66801018 Ki = 46 nM T67162 CBO9U3 66801028 Ki = 33 nM T67162 C3K8DC 66801052 Ki = 4.4 nM T67162 CA4DM3 66801062 Ki = 11 nM T67162 C2OUX9 66801107 Ki = 13 nM T67162 C1H8BS 66801116 Ki > 10000 nM T67162 C4JGC6 66801120 Ki = 23 nM T67162 CX2GN1 66801139 Ki = 36 nM T67162 C1NG8S 66801140 Ki = 39 nM T67162 CR7OW6 66801158 Ki = 15 nM T67162 CJU53X 66801160 Ki = 37 nM T67162 CH3BJ8 66801167 Ki = 4 nM T67162 C0AV5M 66801173 Ki = 15 nM T67162 C0V9EF 66801186 Ki = 15 nM T67162 CTHY41 66801210 Ki = 1.5 nM T67162 CSD67P 66801225 Ki = 22 nM T67162 C8J3YU 66801226 Ki > 10000 nM T67162 CX45OZ 66801229 Ki = 18 nM T67162 C1S0EV 66801230 Ki = 3.2 nM T67162 C7S1KY 66801234 Ki = 3.7 nM T67162 CB53AV 66801246 Ki > 1000 nM T67162 C3F1TZ 66801251 Ki = 27 nM T67162 CF8O9U 66801259 Ki = 170 nM T67162 C2Q9FS 66801263 Ki = 57 nM T67162 C7Y9VP 66801267 Ki > 10000 nM T67162 CED17M 66801271 Ki = 8.7 nM T67162 C41VYW 66801295 Ki = 1.7 nM T67162 C2FYL1 66801333 Ki = 1300 nM T67162 CS75LK 66801335 Ki = 27 nM T67162 CR2N0J 66801344 Ki = 3.7 nM T67162 CDH7S9 66801346 Ki = 14 nM T67162 CGC4U6 66801354 Ki = 7200 nM T67162 CY4FM5 66801379 Ki = 16 nM T67162 C3RX4C 66801425 Ki = 3 nM T67162 C7JD0I 66801429 Ki = 350 nM T67162 CN8OU1 66801430 Ki = 67 nM T67162 C93EGP 66801455 Ki = 46 nM T67162 COR1H8 66801528 Ki = 14 nM T67162 C1F3YV 66801537 Ki = 44 nM T67162 CIRW86 66801551 Ki = 1.9 nM T67162 C75WXP 66801561 Ki = 0.3 nM T67162 C8H5PD 66801565 Ki > 1000 nM T67162 CT5SP8 66801605 Ki = 45 nM T67162 C8MH0I 66801613 Ki = 7.8 nM T67162 CC8JV6 66801624 Ki = 180 nM T67162 C3EI2F 66801625 Ki = 100 nM T67162 C49XBJ 66801673 Ki > 10000 nM T67162 C0XG6B 66801701 Ki = 56 nM T67162 C42EBQ 66801837 Ki = 99 nM T67162 CW3AI2 66803474 Ki = 3.3 nM T67162 CPKH06 66803497 Ki = 5.6 nM T67162 CNJE57 66803500 Ki = 2.5 nM T67162 CN6FZ1 66803595 Ki = 1.5 nM T67162 CREF79 67325096 Ki = 2089.3 nM T67162 CLA7F3 68281136 Ki = 56 nM T67162 C84MZH 68281137 Ki = 400 nM T67162 C5OHR2 68568959 Ki = 2.138 nM T67162 CMI76W 68630558 Ki = 10.47 nM T67162 CD3U6K 68731121 Ki > 10000 nM T67162 C6IP8Q 69082816 Ki > 10000 nM T67162 C34GMW 69599704 Ki = 2700 nM T67162 CQH61C 70681318 Ki = 8.7 nM T67162 CT65MH 70681573 Ki = 9914 nM T67162 C9VL7R 70682090 Ki = 223.61 nM T67162 CT38JR 70683414 Ki = 225 nM T67162 CZ41VT 70683643 Ki = 14.2 nM T67162 C0G2XO 70683685 Ki > 10000 nM T67162 C6PD9Q 70684338 Ki = 38000 nM T67162 CTHV58 70684339 Ki = 16000 nM T67162 COY65E 70684965 Ki = 6.7 nM T67162 CND4A2 70685780 Ki = 3250 nM T67162 C6W9UK 70685781 Ki = 29.7 nM T67162 C2Q6PU 70685835 Ki > 10000 nM T67162 C09VIL 70686262 Ki = 900 nM T67162 CB9V3R 70686493 Ki = 3900 nM T67162 C1P3GF 70686494 Ki = 66000 nM T67162 C3V5QJ 70686495 Ki = 5000 nM T67162 C4REJ6 70687910 Ki = 364 nM T67162 COZN69 70687957 Ki > 1000 nM T67162 C9F7NS 70687958 Ki > 10000 nM T67162 C2U6KV 70688594 Ki = 42000 nM T67162 C4QNS1 70689942 Ki = 4189 nM T67162 C0D7IM 70689943 Ki = 48.6 nM T67162 CY1BV3 70689944 Ki = 8.2 nM T67162 CF7X1W 70690499 Ki = 346.76 nM T67162 CG80JF 70690651 Ki = 12000 nM T67162 CZH6F9 70690652 Ki = 2000 nM T67162 C6TJA5 70690653 Ki = 2000 nM T67162 CPO08R 70691861 Ki > 3800 nM T67162 CD37EI 70691866 Ki = 69 nM T67162 C8YMI5 70692100 Ki = 70.7 nM T67162 C6AUC3 70692138 Ki > 10000 nM T67162 C4A7QI 70692139 Ki > 10000 nM T67162 CN98XB 70692573 Ki = 23000 nM T67162 C9J3TO 70692655 Ki = 146.99 nM T67162 C96FHP 70692656 Ki = 160.99 nM T67162 CU82LJ 70692801 Ki = 7400 nM T67162 C18ETD 70692802 Ki = 12000 nM T67162 C74NGV 70693417 Ki = 15 nM T67162 C6YOS1 70693729 IC50 = 2630.27 nM T67162 CIEG52 70694142 Ki = 69.6 nM T67162 CR7OD5 70694143 Ki = 277.8 nM T67162 C9HV4J 70694144 Ki = 82.4 nM T67162 CU4EK1 70694145 Ki = 201.6 nM T67162 C76JRL 70694146 Ki = 48.7 nM T67162 CQZ38N 70696271 Ki = 482.5 nM T67162 C98YAU 70696888 Ki = 7000 nM T67162 C5U4XV 71109897 Ki = 32 nM T67162 CC43QK 71151588 Ki = 6.3 nM T67162 CG5A0O 71151591 Ki = 21 nM T67162 CB4K3V 71151664 Ki = 95 nM T67162 CO8CB3 71151683 Ki = 45 nM T67162 C5U2BI 71151704 Ki = 23 nM T67162 CU74VQ 71151756 Ki = 120 nM T67162 CVMJ59 71151757 Ki = 78 nM T67162 C4AF8X 71151767 Ki = 11 nM T67162 CN05SR 71151870 Ki = 44 nM T67162 CG18YE 71151889 Ki = 76 nM T67162 CC9M3F 71151924 Ki = 6.1 nM T67162 CP9A6W 71151925 Ki = 62 nM T67162 C2V5SX 71151929 Ki = 47 nM T67162 CM4QC9 71151933 Ki = 1.3 nM T67162 CYP91I 71151953 Ki = 1.3 nM T67162 CN4AJ3 71152026 Ki = 12 nM T67162 C2AQ7H 71195187 Ki > 1000 nM T67162 CON49H 71261649 Ki = 105 nM T67162 CP6B7E 71315272 Ki = 7.943 nM T67162 C0O5KW 71449034 Ki = 6600 nM T67162 C4K5YQ 71449110 Ki > 1000 nM T67162 C91SZN 71449641 Ki = 46 nM T67162 C2GCN7 71449642 Ki = 318 nM T67162 CQN93U 71449643 Ki = 24 nM T67162 CEJ3B4 71449644 Ki = 60 nM T67162 C5SAJ1 71449645 Ki = 25 nM T67162 CSC3R7 71450213 Ki = 1233 nM T67162 CS7M2G 71450549 Ki = 2830 nM T67162 C5IN6O 71450695 Ki = 19 nM T67162 CH3TV9 71450696 Ki = 2002 nM T67162 C97MYL 71450697 Ki = 41 nM T67162 CE6YD5 71450707 Ki = 57 nM T67162 CBP03H 71450812 Ki = 210 nM T67162 C67MOE 71450871 Ki = 3180 nM T67162 CDI84E 71450922 IC50 > 10000 nM T67162 CHT21G 71451454 Ki = 1059 nM T67162 C2QZL4 71451455 Ki = 50 nM T67162 CXI5Q2 71451456 Ki = 76 nM T67162 CKJZ57 71451457 Ki = 16 nM T67162 C0F1HU 71451458 Ki = 36 nM T67162 CTZ24N 71451459 Ki = 20 nM T67162 C70JUP 71451460 Ki = 39 nM T67162 C08KHB 71452040 Ki = 118 nM T67162 C0XW8E 71452041 Ki = 450 nM T67162 C01RKV 71452519 Ki = 803 nM T67162 CK8HN7 71452737 EC50 > 10000 nM T67162 CKI58Z 71453278 Ki = 15 nM T67162 C1QM8D 71453279 Ki = 78 nM T67162 C6O4KT 71453280 Ki = 18 nM T67162 CL49VI 71453281 Ki = 25 nM T67162 CGXT64 71453282 Ki = 8 nM T67162 CN4AJ2 71454274 Ki = 26 nM T67162 CE0R9D 71454275 Ki = 371 nM T67162 C3S5EJ 71454276 Ki = 1535 nM T67162 C4X9KY 71454294 Ki = 92 nM T67162 CA65OQ 71454295 Ki = 17 nM T67162 C8YKT4 71454405 Ki = 92 nM T67162 CFWR57 71454487 Ki = 170 nM T67162 CQMK12 71454927 Ki = 490 nM T67162 CGO13Q 71454997 Ki = 32 nM T67162 C0K1JV 71454998 Ki = 66 nM T67162 C3JF1D 71454999 Ki = 51 nM T67162 C2QZ1N 71455000 Ki = 63 nM T67162 C6FE5D 71455001 Ki = 523 nM T67162 C4L0JN 71455002 Ki = 16 nM T67162 CT2Z8R 71456033 Ki = 27 nM T67162 CD4HQ6 71456045 Ki = 68 nM T67162 CD78KL 71456046 Ki = 140 nM T67162 CZ7XH9 71456235 Ki = 5740 nM T67162 C1H3MD 71456253 EC50 > 10000 nM T67162 CWR40I 71456780 Ki = 560 nM T67162 CZUX67 71456781 Ki = 16 nM T67162 CZ17FC 71456782 Ki = 11 nM T67162 CKF09U 71456783 Ki = 72 nM T67162 CJKV72 71456784 Ki = 10 nM T67162 CNV8U3 71456928 Ki = 235 nM T67162 C7MNB5 71457264 Ki = 302.6 nM T67162 CDSX56 71457372 Ki = 831 nM T67162 C8YD9T 71457837 Ki = 157 nM T67162 CSX5J0 71457844 Ki = 37 nM T67162 CNM83V 71457956 Ki = 310 nM T67162 CNQ5B6 71458040 Ki = 280 nM T67162 C1EA6Q 71458069 Ki = 1000 nM T67162 C84QJC 71458071 Ki = 2400 nM T67162 C37EBC 71458647 Ki = 50 nM T67162 CM6OP1 71458648 Ki = 839 nM T67162 CRGE05 71458649 Ki = 729 nM T67162 CJN4S1 71458650 Ki = 67 nM T67162 CNT5J9 71458651 Ki = 10 nM T67162 C3NAM7 71458652 Ki = 41 nM T67162 C3X1ZG 71459659 EC50 = 1.7 nM T67162 CH5YG1 71459660 EC50 = 0.44 nM T67162 CI6OW4 71459759 Ki = 65 nM T67162 CSY3U1 71459760 Ki = 60 nM T67162 CD10CQ 71459761 Ki = 95 nM T67162 CYGO39 71459901 Ki = 19.95 nM T67162 CG0WO9 71459954 Ki > 2000 nM T67162 CT17XB 71460468 Ki = 79 nM T67162 CAT73U 71460601 EC50 = 50 nM T67162 C9ESJ4 71461481 Ki = 76 nM T67162 C9VE0P 71462090 Ki = 160 nM T67162 C7AX1Q 71462178 Ki = 24 nM T67162 C1CS0Z 71462179 Ki = 72 nM T67162 CUG7M5 71463194 Ki = 187 nM T67162 C1XUO3 71463195 Ki = 10820 nM T67162 C7IE9K 71463196 Ki = 12160 nM T67162 C6EF4I 71463197 Ki = 574 nM T67162 C82GIQ 71463207 Ki = 8.3 nM T67162 CD64WC 71500036 Ki = 15 nM T67162 C1E9HB 71502591 Ki = 20 nM T67162 CE9ZL1 71502631 Ki = 290 nM T67162 CQ3EZ2 71502632 Ki = 67 nM T67162 CQ8FW4 71502633 Ki = 110 nM T67162 CBY90L 71502676 Ki = 220 nM T67162 CTA3J9 71508640 Ki = 15 nM T67162 C82BQI 71508682 Ki = 880 nM T67162 C93CKS 71508683 Ki = 150 nM T67162 C5TM0Z 71508684 Ki = 6400 nM T67162 CSI68J 71508685 Ki = 27 nM T67162 CC8O1Y 71508686 Ki = 260 nM T67162 CPW6F5 71508687 Ki = 76 nM T67162 CC2R3L 71508710 Ki = 1100 nM T67162 CMJQ82 71508711 Ki = 830 nM T67162 CN43VA 71508712 Ki = 220 nM T67162 CNM08F 71508713 Ki = 160 nM T67162 CQ2N0J 71508866 IC50 = 7960 nM T67162 C2VP0I 71528204 EC50 = 1.4 nM T67162 CE92DF 71528209 Ki = 1971 nM T67162 CK2EY7 71540967 Ki = 3900 nM T67162 C3WR0T 71541076 IC50 = 1400 nM T67162 C0SKF2 71541077 Ki = 2500 nM T67162 C45CNE 71541078 Ki = 1100 nM T67162 C3UR6G 71541079 Ki = 5000 nM T67162 CQ0D2T 71541080 Ki = 5000 nM T67162 C9VF1X 71541081 Ki = 800 nM T67162 CBN7X9 71541082 Ki = 4300 nM T67162 CJ89BQ 71541083 Ki = 80 nM T67162 C9T1HK 71541084 Ki = 75 nM T67162 C4PYZ6 71541174 Ki = 42 nM T67162 C1RZ5T 71541175 Ki = 92 nM T67162 CF1B8U 71541176 Ki = 34 nM T67162 CU5E7L 71541177 Ki = 42 nM T67162 C9I1QA 71541178 Ki = 42 nM T67162 CA5O1N 71541179 Ki = 5000 nM T67162 CZUV57 71541180 Ki = 200 nM T67162 CXS47M 71541275 Ki = 38 nM T67162 C3AFY4 71541276 Ki = 320 nM T67162 C98TJN 71541277 Ki = 490 nM T67162 C4AG9L 71541278 Ki = 580 nM T67162 CVX93I 71541279 Ki = 5000 nM T67162 C1J4KM 71541280 Ki = 350 nM T67162 CWQ5R6 71562963 Ki = 101 nM T67162 CG1ZU7 71562964 Ki = 14.8 nM T67162 CI3EW5 71562965 Ki > 10000 nM T67162 C51IHJ 71562966 Ki = 195 nM T67162 CW2V1F 71563082 Ki = 132 nM T67162 C4ZKF0 71563083 Ki = 12.3 nM T67162 CR8UF1 71563084 Ki = 4 nM T67162 CJ34IH 71571360 IC50 > 50000 nM T67162 C5PHM9 71571370 IC50 > 100000 nM T67162 CS0FY1 71571378 IC50 = 6000 nM T67162 CUN24P 71571394 IC50 = 9000 nM T67162 CDU24A 71571402 IC50 = 9600 nM T67162 C83LQO 71571413 IC50 > 50000 nM T67162 CC02ZH 71571419 IC50 > 50000 nM T67162 C0M7QU 71571423 IC50 > 10000 nM T67162 C1Z2OC 71571433 IC50 = 6800 nM T67162 CRMC90 71571436 IC50 > 50000 nM T67162 CT2ME3 71574204 Ki = 8 nM T67162 C62RWV 71574210 Ki = 16 nM T67162 CKC53S 71574212 Ki = 9 nM T67162 C2LXH5 71574302 Ki = 11 nM T67162 CK7GM0 71574306 Ki = 17 nM T67162 CO3E4N 71583848 Ki = 33 nM T67162 C8N2ML 71583849 Ki = 28 nM T67162 CO4P6L 71604368 EC50 = 2900 nM T67162 C6W5AU 71604371 IC50 = 18000 nM T67162 CWAO49 71604376 EC50 = 2300 nM T67162 CN9ST4 71604379 IC50 > 50000 nM T67162 CJCO20 71604380 IC50 > 100000 nM T67162 CVDZ96 71653289 Ki = 3800 nM T67162 C1NDY0 71653447 Ki = 580 nM T67162 CZ0DB6 71653589 Ki = 1500 nM T67162 C04CZK 71653734 Ki = 12 nM T67162 C5VH2Z 71657942 Ki = 119 nM T67162 CY9ES0 71657943 Ki = 101 nM T67162 CU41CZ 71657944 Ki = 125 nM T67162 C0S6YV 71657945 Ki = 108 nM T67162 CX52VK 71657946 Ki = 128 nM T67162 C6KJW5 71657947 Ki = 111 nM T67162 C6AQG0 71658072 Ki = 95.2 nM T67162 CQ3W7X 71658073 Ki = 56.5 nM T67162 CE3V4J 71658074 Ki = 138 nM T67162 C40XRK 71658075 Ki = 125 nM T67162 CPI8E9 71658076 Ki = 107 nM T67162 CC1U6V 71658077 Ki = 151 nM T67162 C8LX4D 71658203 Ki = 100 nM T67162 CVX3G1 71658204 Ki = 43.7 nM T67162 C29STX 71658205 Ki = 280 nM T67162 CR0EN8 71658206 Ki = 119 nM T67162 CF41PZ 71658207 Ki = 145 nM T67162 C7LMV3 71658208 Ki = 152 nM T67162 CIAR53 71658338 Ki = 169 nM T67162 CZ65JA 71659909 Ki = 128 nM T67162 C8PLQ7 71660285 EC50 = 179 nM T67162 CI0GU8 71660496 IC50 > 48500 nM T67162 C50YDS 71716758 IC50 > 10000 nM T67162 C65JRT 71717830 IC50 = 2420 nM T67162 CGU06V 71717958 IC50 > 10000 nM T67162 CW35XI 71722291 EC50 = 76 nM T67162 C4EC8K 71722293 EC50 = 5.1 nM T67162 C4FJV9 71722295 EC50 = 49 nM T67162 C8H5OT 71722297 EC50 = 3.4 nM T67162 C3SDV1 71722299 EC50 = 2.7 nM T67162 CY4NH1 71722300 Ki = 79 nM T67162 CTI15V 71724940 EC50 = 800 nM T67162 CGH7I1 71724941 EC50 = 7100 nM T67162 C24SVN 71724943 EC50 = 617 nM T67162 C64GLV 71724944 EC50 = 183 nM T67162 CB3WQ5 71724946 EC50 = 128 nM T67162 CG34PQ 71724947 EC50 = 6200 nM T67162 CF0TW3 71724948 EC50 = 7800 nM T67162 CV5OH2 71724949 EC50 = 5500 nM T67162 CKP3M7 71724951 EC50 = 1700 nM T67162 CUB76P 71724952 EC50 = 180 nM T67162 CE4A7V 71724954 IC50 > 50000 nM T67162 CD53XP 71724955 EC50 = 5200 nM T67162 CLTX37 71724956 IC50 > 50000 nM T67162 C4YA9Q 71724957 EC50 = 1100 nM T67162 C9C2IE 71724959 EC50 = 217 nM T67162 CDW76R 71724960 EC50 = 4600 nM T67162 C1BYT9 71724961 EC50 = 13000 nM T67162 C3TAK6 71724962 EC50 = 6000 nM T67162 CI0D9X 71724963 EC50 = 4200 nM T67162 C2I1ML 71724964 EC50 = 364 nM T67162 C9P2RK 71724965 EC50 = 2500 nM T67162 C0X8AZ 71724966 EC50 = 2400 nM T67162 CBIF31 71724967 EC50 = 617 nM T67162 C2LI5P 71724968 EC50 = 3000 nM T67162 CH6C3U 71724969 EC50 > 50000 nM T67162 CI3V7S 71724970 EC50 = 1800 nM T67162 CC08MW 71724971 EC50 = 210 nM T67162 CZIH39 71724974 EC50 = 6100 nM T67162 CD2U5X 71724975 EC50 = 4100 nM T67162 CPIC98 71724976 EC50 = 786 nM T67162 CXM9B5 71724977 EC50 = 7800 nM T67162 CM63QP 71724978 EC50 = 2600 nM T67162 C6C9IT 71724979 EC50 > 100000 nM T67162 CQRY07 71724980 EC50 = 1400 nM T67162 CJS8I1 71724983 EC50 > 100000 nM T67162 CC7T2D 71724985 EC50 = 1300 nM T67162 CC5FG2 71724986 EC50 = 4300 nM T67162 CV09TJ 71724987 EC50 = 570 nM T67162 CIX5F7 71724989 EC50 = 413 nM T67162 C14LXP 71724991 EC50 = 4400 nM T67162 CUFB92 71724993 EC50 = 10100 nM T67162 CFS28E 71724994 EC50 = 2300 nM T67162 C0F2WP 71724995 EC50 = 138 nM T67162 CEJ2L9 71724996 EC50 = 780 nM T67162 C4NIK3 71725006 IC50 > 100000 nM T67162 CM31ZP 71725009 IC50 > 100000 nM T67162 C8HQP2 71725014 IC50 > 100000 nM T67162 CR6JF2 71725020 IC50 = 9700 nM T67162 C0X4CR 71725021 IC50 > 100000 nM T67162 C2NX3A 71725023 IC50 > 100000 nM T67162 C6MTL4 71725024 IC50 > 10000 nM T67162 C8URA5 71725025 IC50 = 2800 nM T67162 CFY64I 71725026 IC50 > 50000 nM T67162 C09ZBK 71725027 IC50 = 13000 nM T67162 CEZN65 71725031 EC50 = 1700 nM T67162 CXA9N4 71725039 EC50 = 7000 nM T67162 CZ2MG4 71725047 EC50 = 790 nM T67162 C5MH0U 71725048 IC50 > 100000 nM T67162 C54VLH 71725049 IC50 = 3800 nM T67162 C3V6XP 71725052 EC50 = 660 nM T67162 CRV8K6 71725061 EC50 = 4400 nM T67162 CEQL80 71725064 EC50 = 830 nM T67162 C7HKL3 71725065 IC50 = 440 nM T67162 CQO30I 71733932 Ki = 0.6 nM T67162 C93QMB 71733935 Ki = 1.2 nM T67162 COM72V 71734028 Ki = 5.5 nM T67162 C4S5WD 71734029 Ki = 0.55 nM T67162 C2ZX1W 71734031 Ki = 3.1 nM T67162 C7GDW5 71734126 Ki = 3.9 nM T67162 CQJ8P4 71734127 Ki = 1.1 nM T67162 CR53GT 71734129 Ki = 2 nM T67162 CU5R1S 71758594 Ki = 87.3 nM T67162 CF01OQ 71937057 Ki = 1606 nM T67162 C0PSF9 72138721 Ki = 37 nM T67162 CR3Z1P 72152555 Ki = 53 nM T67162 C24ZSV 72152556 Ki = 3420 nM T67162 CWT8O4 72152557 Ki = 2187 nM T67162 CZ49CG 72152558 Ki > 10000 nM T67162 C31THM 72164180 Ki = 1545 nM T67162 C56VLM 72164181 Ki > 10000 nM T67162 CD8A9K 72164182 Ki = 1593 nM T67162 C4C0BH 72164183 Ki = 2167 nM T67162 CQU81Y 72164299 Ki = 327 nM T67162 CF0H7K 72164300 Ki = 351 nM T67162 C7WM5U 72164301 Ki = 242 nM T67162 C4HO2U 72164302 Ki = 502 nM T67162 C08NOR 72187659 EC50 = 1900 nM T67162 CQ70NJ 72187662 EC50 = 3300 nM T67162 CCL54H 72187663 IC50 = 18000 nM T67162 CMPS48 72190766 Ki = 137 nM T67162 C4E8TR 72191064 Ki = 226.6 nM T67162 C85FKU 72191065 Ki = 211.7 nM T67162 CNPA07 72191066 Ki = 198.8 nM T67162 CQL1T2 72191067 Ki = 181.5 nM T67162 CI2M7H 72191068 Ki = 136.6 nM T67162 C3ATN5 72197484 IC50 = 146.7 nM T67162 C20HSN 72197485 IC50 = 63.3 nM T67162 CN8A5R 72197486 IC50 = 85.8 nM T67162 CL3BF7 72197668 IC50 = 162.8 nM T67162 CUVJ59 72197845 Ki = 14 nM T67162 CIKU20 72198011 Ki = 161 nM T67162 COH95V 72198014 Ki = 343 nM T67162 C0WY2V 72198191 Ki = 80 nM T67162 C7AOY4 72198754 IC50 = 3.5 nM T67162 C4M7KP 72198756 IC50 > 100 nM T67162 C0U5RS 72544566 Ki = 460 nM T67162 CVY4I0 72544787 Ki = 1500 nM T67162 C8UM5H 72544789 Ki = 750 nM T67162 CVU61Z 72545007 Ki = 3400 nM T67162 CR6HY3 72545008 Ki = 4700 nM T67162 CC25RP 72545009 Ki = 23000 nM T67162 CW9OZ7 72545010 Ki = 24000 nM T67162 C14DJV 72545011 Ki = 1600 nM T67162 C4E5ZF 72545238 Ki = 340 nM T67162 CY7J8U 72545239 Ki = 2700 nM T67162 CU72QA 72545240 Ki = 440 nM T67162 CWH6T3 72548703 IC50 = 1.8 nM T67162 C4AS0E 72699528 Ki = 8.9 nM T67162 CO20CN 72699532 Ki = 0.35 nM T67162 C8EVJ6 72699690 Ki = 0.42 nM T67162 CEAK86 72699692 Ki = 0.53 nM T67162 CIR7G1 72699716 Ki = 7.54 nM T67162 C9Y3DG 72699717 Ki = 46.7 nM T67162 CRMC07 72699718 Ki = 34.23 nM T67162 COH4F8 72699779 Ki = 2.2 nM T67162 C4X9AO 72699812 Ki = 40.83 nM T67162 C70PWS 72699813 Ki = 79.54 nM T67162 C5K9JW 72699815 Ki = 34.36 nM T67162 CZV6D5 72699816 Ki = 38.63 nM T67162 CIDS43 72699817 Ki = 17.61 nM T67162 C6J8GM 72699818 Ki = 11.51 nM T67162 CC8PL5 72699903 Ki = 16.49 nM T67162 C7YTK9 72699904 Ki = 12.02 nM T67162 C26STM 72700473 Ki = 25 nM T67162 CL96GC 72700475 Ki = 1.7 nM T67162 C45JKS 72700476 Ki = 0.94 nM T67162 C3TO8B 72700557 Ki = 0.33 nM T67162 CVA2X7 72700634 Ki = 0.85 nM T67162 C7W4RH 72734860 Ki = 1400 nM T67162 CK07MC 72735990 EC50 = 33 nM T67162 C39JTD 72735991 Ki = 380.19 nM T67162 C8O2XW 72736197 EC50 = 54 nM T67162 C5VD9Y 72736198 Ki = 23.44 nM T67162 CG1VR4 72736199 EC50 = 144 nM T67162 CM5A8N 72736200 EC50 = 74 nM T67162 C0JAO6 72736201 Ki = 5248.07 nM T67162 CWT25A 72736202 Ki = 912.01 nM T67162 CA9CY1 72736203 EC50 = 12 nM T67162 C5DIN9 72736378 Ki = 245.47 nM T67162 C5HXV6 72736379 Ki = 354.81 nM T67162 CH20UW 72736380 Ki = 1148.15 nM T67162 C1S6DZ 72736381 Ki = 549.54 nM T67162 CGQ63P 72736382 Ki = 309.03 nM T67162 C78FKX 72736383 Ki = 147.91 nM T67162 C7R8EK 72736555 Ki = 42.66 nM T67162 CC01EJ 72737728 IC50 = 16500 nM T67162 C6XYJ3 72737730 Ki = 5500 nM T67162 C6IF9H 72737744 Ki = 5500 nM T67162 CC65OA 73213195 Ki > 10000 nM T67162 CW83DK 73213196 Ki > 10000 nM T67162 CCV91B 73346042 Ki = 37.1 nM T67162 CI8D5O 73346333 Ki > 10000 nM T67162 CK0HR9 73346334 Ki > 10000 nM T67162 C5QYH1 73347474 Ki = 0.53 nM T67162 CY60RD 73347826 Ki = 9906 nM T67162 CQH3J5 73349358 Ki > 10000 nM T67162 C6BS5L 73349361 Ki = 5096 nM T67162 CPN5T8 73350334 IC50 = 870 nM T67162 C9NAE5 73350335 IC50 > 1000 nM T67162 CPZT87 73352849 Ki = 158.49 nM T67162 CCIT57 73353534 Ki = 4.2 nM T67162 C7IA8U 73354844 IC50 > 1000 nM T67162 CX4Q3F 73354845 IC50 = 650 nM T67162 C4F7VK 73355415 Ki = 5675 nM T67162 CO1VP6 73356382 IC50 > 1000 nM T67162 CX17VZ 73670899 IC50 > 500 nM T67162 CG21OC 73671061 Ki = 809 nM T67162 CS82XC 73671062 Ki = 337 nM T67162 CKW82D 73671216 IC50 = 37 nM T67162 CU5S6G 73671217 IC50 = 25 nM T67162 C7AJU1 73671218 Ki = 655 nM T67162 CL4F9C 73671219 IC50 = 161 nM T67162 CLS83G 73671367 Ki = 1883 nM T67162 CUB97Z 74538690 Ki = 345 nM T67162 C2E7QW 75201901 Ki = 8300 nM T67162 C8IDL3 75306277 Ki = 125.89 nM T67162 C45OSP 76284193 Ki = 2450 nM T67162 CS3HT5 76309671 Ki = 28.18 nM T67162 C69BJY 76310154 Ki = 37.15 nM T67162 CN52QU 76310158 Ki = 50.12 nM T67162 C5OYN0 76311261 Ki = 23.9 nM T67162 C2VAS4 76311270 Ki = 42.4 nM T67162 CX40CG 76311272 Ki = 40.4 nM T67162 CPNJ32 76311289 EC50 = 266 nM T67162 CTV52G 76313854 Ki = 50.12 nM T67162 CP40AM 76313855 Ki = 32.36 nM T67162 C3B8FS 76313862 Ki = 41.69 nM T67162 CL8N5U 76314097 IC50 = 16280 nM T67162 C8QJ2B 76314861 Ki = 7.5 nM T67162 C3K1QZ 76314884 EC50 = 224 nM T67162 CQP0O8 76317383 Ki = 645.65 nM T67162 CV6T1W 76317649 IC50 > 30000 nM T67162 CI9Z6N 76317651 IC50 > 30000 nM T67162 CQM65S 76318472 Ki = 120 nM T67162 CX9ON0 76318474 Ki = 5.1 nM T67162 CGZP35 76318476 Ki = 15.7 nM T67162 C2NXG0 76321107 Ki = 46.77 nM T67162 C81DZU 76321374 IC50 > 26000 nM T67162 CIB40D 76321554 EC50 = 0.631 nM T67162 CS9F1X 76321556 EC50 = 1.585 nM T67162 CJH2U5 76322139 Ki = 155 nM T67162 CG4EX6 76322141 Ki = 11.7 nM T67162 C1F3GE 76322158 EC50 = 149 nM T67162 CU73JS 76322159 EC50 = 79 nM T67162 CNA60Z 76322160 EC50 = 248 nM T67162 CW7RV4 76324757 Ki > 10000 nM T67162 CQ8D4Y 76324758 Ki = 19.05 nM T67162 C97LOB 76325150 EC50 = 0.03162 nM T67162 CCR29U 76325152 EC50 = 0.3981 nM T67162 C6GBK1 76325154 Ki = 144.54 nM T67162 CLP59V 76325156 EC50 = 0.05012 nM T67162 C3K6UP 76325763 Ki = 119 nM T67162 CB8O1P 76325786 EC50 = 396 nM T67162 C8SOZ7 76328295 Ki = 120.23 nM T67162 C5M8OD 76328296 Ki = 87.1 nM T67162 C2O0FW 76328713 Ki = 0.1622 nM T67162 C17YTI 76328715 EC50 = 0.1585 nM T67162 C97XIE 76329028 EC50 = 36.8 nM T67162 C0ED1J 76329346 Ki = 33.6 nM T67162 CRSK62 76329369 EC50 = 110 nM T67162 C5L2NC 76329370 EC50 = 385 nM T67162 CTL3I7 76331989 Ki = 17.38 nM T67162 CDM84V 76332211 IC50 > 30000 nM T67162 CL2N3Y 76332978 Ki = 21.8 nM T67162 CC16RS 76332985 Ki = 66.3 nM T67162 CLJ16D 76332987 Ki = 60 nM T67162 CV1O9C 76332989 Ki = 2 nM T67162 CEI18J 76333011 EC50 = 419 nM T67162 CGBE87 76335066 Ki = 51.3 nM T67162 CZFD79 76335466 EC50 = 0.17 nM T67162 CUO0S5 76335562 Ki = 112.2 nM T67162 CL41EG 76335563 Ki = 177.83 nM T67162 C67EJQ 76335845 IC50 > 30000 nM T67162 CL2I3A 76336596 Ki = 5.9 nM T67162 CA6YD8 76336623 EC50 = 10 nM T67162 CK45CZ 76336624 EC50 = 132 nM T67162 C1UZ5J 76441180 Ki = 37.7 nM T67162 C28RIZ 76518514 Ki = 33 nM T67162 CWI52H 77974401 Ki > 1000 nM T67162 CWG4T2 78209992 IC50 = 797 nM T67162 CEAC35 85469680 EC50 = 13 nM T67162 C5JH2Y 85470564 EC50 = 45 nM T67162 C8EWX5 85658088 Ki = 2877 nM T67162 CQ9H4U 86277844 IC50 > 10000 nM T67162 CJ9N5Q 86280005 Ki = 15.8 nM T67162 CEPC94 86288948 Ki = 715 nM T67162 CUA89I 86341962 Ki = 0.71 nM T67162 CWPH45 86341996 Ki = 0.63 nM T67162 CCR8X7 86342061 Ki = 0.51 nM T67162 CY2I8J 86342094 Ki = 2.4 nM T67162 CC47HJ 86342098 Ki = 1.4 nM T67162 CK03YC 86342156 Ki = 2.9 nM T67162 C5AQK2 86342192 Ki = 0.19 nM T67162 C9DZ2I 86342193 Ki = 0.21 nM T67162 CQP38R 86342194 Ki = 0.43 nM T67162 CE39OD 86342294 Ki = 0.43 nM T67162 CHE2U4 90178632 Ki = 631 nM T67162 CD7R6P 90213677 Ki = 4.6 nM T67162 CT8HK6 90389439 Ki = 693 nM T67162 CU9ED1 90389592 Ki = 298 nM T67162 CU8L2K 90466425 EC50 = 56.4 nM T67162 CIM5O2 90466573 EC50 = 39.9 nM T67162 CFDK42 90466574 EC50 = 13 nM T67162 C1HQP6 90466717 EC50 = 21.5 nM T67162 C5GX4U 90466867 EC50 = 147 nM T67162 C82YRS 90467020 EC50 = 66.2 nM T67162 C6B8ZY 90467021 EC50 = 13.7 nM T67162 CT0N3V 90467024 EC50 = 54.2 nM T67162 CB61FX 90467322 EC50 = 57.9 nM T67162 C8C1KA 90467323 EC50 = 10.4 nM T67162 CYUQ73 90467453 EC50 = 49.3 nM T67162 C5EN3B 90643433 Ki > 1000 nM T67162 CH01QM 90643434 Ki > 1000 nM T67162 CB6I7A 90643699 Ki = 1220 nM T67162 C3EY5T 90643700 Ki = 923 nM T67162 CKYP81 90643701 Ki = 667 nM T67162 CF5U1L 90643702 Ki = 623 nM T67162 C80SXV 90644057 Ki = 1092 nM T67162 C20EPB 90644058 Ki = 1543 nM T67162 C04MRN 90644059 Ki > 10000 nM T67162 CIA8J4 90644060 Ki = 1417 nM T67162 CY8TP0 90644061 Ki = 1046 nM T67162 CKV24H 90644062 Ki = 1000 nM T67162 CW2ZC4 90644063 Ki = 1861 nM T67162 CLG60I 90644064 Ki = 3108 nM T67162 CKLN72 90644065 Ki = 3962 nM T67162 C7G5VH 90644066 Ki = 1979 nM T67162 CLM0J5 90644067 Ki = 630.96 nM T67162 CDPE48 90644071 Ki = 2507 nM T67162 CFDW68 90644074 Ki = 2000 nM T67162 C0T8RE 90644075 Ki = 63 nM T67162 C2KE9G 90644076 Ki = 55 nM T67162 C1SOF5 90644077 Ki = 15 nM T67162 CIE9Z2 90644078 Ki = 30 nM T67162 CLFV10 90644226 Ki = 6.7 nM T67162 CZ7LD8 90644227 Ki = 2.3 nM T67162 C35GPQ 90644228 Ki = 14 nM T67162 CZI30L 90644230 Ki = 6.7 nM T67162 CUO0J6 90644928 Ki = 800 nM T67162 CF9HI4 90644929 Ki = 2500 nM T67162 CX2WE7 90644930 Ki = 7400 nM T67162 C2YUK1 90645287 Ki = 42.6 nM T67162 C56CJM 90645288 Ki = 15.49 nM T67162 CFA45E 90645289 EC50 = 0.3 nM T67162 CB06RP 90645290 Ki = 9.1 nM T67162 CBF6I0 90645291 Ki = 2750 nM T67162 CGO87K 90645292 Ki = 1348.96 nM T67162 CQ1E9A 90645293 Ki = 2089.3 nM T67162 C17LOB 90645294 Ki = 2041.74 nM T67162 CP2G4B 90645295 Ki = 891.25 nM T67162 C2R3IT 90645296 IC50 = 93.33 nM T67162 C6NG9T 90645297 EC50 = 1.43 nM T67162 C0HIN1 90645298 IC50 = 3.98 nM T67162 COV1T8 90645299 Ki = 910 nM T67162 CLD0X8 90645300 Ki = 1698.24 nM T67162 C9B0SM 90645301 Ki = 2238.72 nM T67162 C2T3LB 90645302 Ki = 1980 nM T67162 C2MOX7 90645303 Ki = 975 nM T67162 C04SZK 90645304 Ki = 47.86 nM T67162 CDV07H 90645305 Ki = 19.5 nM T67162 C1V8HN 90645306 Ki = 6.3 nM T67162 C95GZE 90645307 EC50 = 2.69 nM T67162 CRV91A 90645308 Ki = 0.6 nM T67162 CVY38R 90656834 Ki = 0.63 nM T67162 CYW9H7 90656835 Ki = 21.47 nM T67162 C8Y4ZV 90656836 Ki = 9.69 nM T67162 CE8PX9 90656837 Ki = 10.32 nM T67162 CC9IO3 90656838 Ki = 27.32 nM T67162 C7N1ZB 90656839 Ki = 12.27 nM T67162 CVM5N8 90656840 Ki = 8.14 nM T67162 CTN27W 90656841 Ki = 12.96 nM T67162 C9HZU8 90656842 Ki = 8.01 nM T67162 CJ9TM7 90656843 Ki = 28.43 nM T67162 C1YV6C 90656844 Ki = 30.33 nM T67162 CW0F8X 90656845 Ki = 23.78 nM T67162 CGCE27 90656846 Ki = 1.47 nM T67162 C8VCJ9 90656847 Ki = 27.39 nM T67162 CM7R6L 90656848 Ki = 53.92 nM T67162 C63WZB 90656849 Ki = 25.27 nM T67162 C56LVY 90656850 Ki = 26.13 nM T67162 C9A7KB 90656851 Ki = 35.77 nM T67162 CY2BQ0 90656852 Ki = 42.8 nM T67162 CKB09V 90656853 Ki = 44.67 nM T67162 CCG37D 90656854 Ki = 5.98 nM T67162 CTC5M6 90656855 Ki = 52.03 nM T67162 C4KCA8 90656856 Ki = 64.16 nM T67162 C1JF7H 90656857 Ki = 7.31 nM T67162 CDJ7B0 90656858 Ki > 1000 nM T67162 C4MUI2 90664601 IC50 = 1369 nM T67162 CHT7D5 90664962 IC50 = 908 nM T67162 C9JQ8U 90666896 Ki = 63.1 nM T67162 CVI58C 90666898 Ki = 32.36 nM T67162 CACG19 90666899 Ki = 199.53 nM T67162 C4HPT5 90666900 Ki = 173.78 nM T67162 C86HDZ 90666902 Ki = 199.53 nM T67162 CODM50 90666903 Ki = 158.49 nM T67162 CSN13Z 90666904 Ki = 54.95 nM T67162 CP7HX3 90667734 Ki = 3.9 nM T67162 CNB56Y 90899701 IC50 = 76 nM T67162 CSRU41 91242334 IC50 = 131 nM T67162 CB3SW9 91379597 Ki = 61.66 nM T67162 C0J5YH 91864602 Ki = 125.89 nM T67162 CRX16J 91884611 IC50 = 3.31 nM T67162 C3K4LU 91937908 Ki = 219 nM T67162 C3S6VX 92209551 IC50 = 1.1 nM T67162 CCV0I4 92640710 Ki > 100000 nM T67162 CLR87F 94496003 Ki = 334 nM T67162 CNUM64 95104704 Ki = 1996 nM T67162 CK83CL 95198280 Ki = 1522 nM T67162 CMG1N3 95214051 Ki = 4918 nM T67162 C5GJA7 95232163 Ki = 7745 nM T67162 C8QJW7 95338888 Ki = 5044 nM T67162 C0BAG2 95339350 Ki = 6912 nM T67162 C4BRK3 95339542 Ki = 3129 nM T67162 C8XFV3 101007561 Ki = 42.66 nM T67162 CC02RF 101885473 EC50 = 22 nM T67162 C2HJC5 101885474 EC50 = 28 nM T67162 C1BL9H 101885475 EC50 = 3.89 nM T67162 CX06ZV 101885476 EC50 = 14 nM T67162 CK4EM7 101885477 EC50 = 6.166 nM T67162 COA3U6 102262219 Ki = 3200 nM T67162 CE6Z3M 109030343 EC50 = 154 nM T67162 CC1P6O 109030515 Ki = 1490 nM T67162 CP6F4D 112815120 Ki = 71.9 nM T67162 CTYH92 117028759 Ki = 99379 nM T67162 C1ZBQ9 117365679 EC50 > 100000 nM T67162 C7P5RX 117869686 IC50 = 248 nM T67162 C59ZAJ 117870140 Ki = 176 nM T67162 CS8YG9 117870408 Ki = 361 nM T67162 CJ7KU8 117870413 Ki = 13567 nM T67162 C95QKZ 117870490 Ki = 366 nM T67162 CU5S8B 117870714 Ki = 4604 nM T67162 CNM0U7 117870915 Ki = 4983 nM T67162 CV80LK 117870976 Ki = 934 nM T67162 C5I4TZ 117871054 Ki = 191 nM T67162 C5HR9I 117871069 Ki = 72 nM T67162 C1KDN4 117871083 Ki = 1452 nM T67162 CIK45N 117949627 Ki = 88.02 nM T67162 CSH7K4 117949705 Ki = 18.38 nM T67162 CMSN80 118626035 Ki = 16 nM T67162 CT3AI0 118626042 Ki = 37 nM T67162 CKNJ72 118626045 Ki = 5 nM T67162 CGB42Y 118626088 Ki = 12 nM T67162 C0XJT5 118626089 Ki = 11 nM T67162 CIE4C7 118626101 Ki = 3 nM T67162 C1NYS5 118626120 Ki = 19 nM T67162 CPG04R 118626121 Ki = 5 nM T67162 C3S5LJ 118626129 Ki = 4 nM T67162 CY3F0N 118626140 Ki = 13 nM T67162 CE07IQ 118626142 Ki = 6 nM T67162 C72OZY 118626161 Ki = 0.7 nM T67162 CY3E7S 118626169 Ki = 22 nM T67162 CHRB75 118626208 Ki = 13 nM T67162 C2I0HB 118643968 Ki = 78.6 nM T67162 CJS6B2 118709159 Ki = 5.4 nM T67162 C9XDM6 118709160 Ki = 12 nM T67162 CQ9C5S 118709161 Ki = 2.3 nM T67162 C1YRW4 118709162 Ki = 2.6 nM T67162 CPL69Z 118709163 Ki = 2.5 nM T67162 CGAB49 118709164 Ki = 5.6 nM T67162 C3SX4Z 118709165 Ki = 15 nM T67162 CC7FW6 118709166 Ki = 46 nM T67162 CRMK67 118709167 Ki = 62 nM T67162 CW4YS6 118709168 Ki = 140 nM T67162 CY3BR2 118709169 Ki = 150 nM T67162 CIX72C 118709170 Ki = 25 nM T67162 C2O8BG 118709171 Ki = 280 nM T67162 COV8K7 118709172 Ki = 47 nM T67162 CJZD82 118709173 Ki = 1.1 nM T67162 C16WQU 118709174 Ki = 2.2 nM T67162 C4E5MK 118709175 Ki = 1.8 nM T67162 CFV2M0 118709176 Ki = 1.3 nM T67162 C08TAX 118709177 Ki = 4.9 nM T67162 CYNM75 118709178 Ki = 1 nM T67162 CJZ7G0 118709179 Ki = 1.6 nM T67162 CSB25E 118709750 Ki = 27 nM T67162 CD4S9R 118709751 Ki = 4.8 nM T67162 CBG0D4 118710458 Ki = 178 nM T67162 CR90MQ 118710459 Ki = 12 nM T67162 CN9HD5 118710460 IC50 = 60 nM T67162 C13SFN 118710461 Ki = 191 nM T67162 CIWT51 118710462 Ki = 1303 nM T67162 CZ2HV3 118710463 Ki = 1563 nM T67162 CW1I6Z 118710464 Ki = 24938 nM T67162 CW14NI 118710465 Ki = 3646 nM T67162 CZ7WQ3 118710466 IC50 = 418 nM T67162 CK2XE7 118710467 IC50 = 301 nM T67162 CFBT50 118710468 Ki = 683 nM T67162 CR97VN 118710469 Ki = 481 nM T67162 C9CJ5R 118710470 IC50 = 311 nM T67162 CO8E9F 118711252 Ki > 1000 nM T67162 CJY9D7 118711253 Ki > 1000 nM T67162 CFJE45 118711254 Ki > 1000 nM T67162 CK1A2W 118711255 Ki > 1000 nM T67162 CNQJ96 118711256 Ki > 1000 nM T67162 CJ91QY 118711257 Ki > 1000 nM T67162 C42YEC 118711258 Ki > 1000 nM T67162 CU6BT0 118711259 Ki > 1000 nM T67162 C97RTC 118711260 Ki > 1000 nM T67162 CM47VI 118711261 Ki > 1000 nM T67162 CX3M2Z 118711262 Ki > 1000 nM T67162 CN59OU 118711263 Ki > 1000 nM T67162 CXI0S9 118711264 Ki > 1000 nM T67162 CW3F4T 118711265 Ki > 1000 nM T67162 C4UAV9 118711266 Ki > 1000 nM T67162 C83MBF 118711267 Ki > 1000 nM T67162 C9FH2L 118711268 Ki > 1000 nM T67162 CBP47E 118711269 Ki > 1000 nM T67162 C7W2QM 118711270 Ki > 1000 nM T67162 C6QS7R 118711271 Ki > 1000 nM T67162 C6ZF8M 118711272 Ki > 1000 nM T67162 CDP7I9 118711273 Ki > 1000 nM T67162 CAF7I0 118711274 Ki > 1000 nM T67162 C4R3NA 118714496 Ki = 30 nM T67162 C8AUL2 118714497 Ki = 5.4 nM T67162 CW8F2K 118714498 Ki = 37 nM T67162 CE89TI 118714552 IC50 = 16500 nM T67162 C5LFW4 118717221 Ki > 1000 nM T67162 CK98PG 118717796 Ki = 29.1 nM T67162 C43TKI 118717797 Ki = 189.99 nM T67162 CE5M8O 118719791 Ki = 64 nM T67162 C8M1VO 118719792 Ki = 30.9 nM T67162 CQY62K 118719793 Ki = 19.4 nM T67162 C97UXN 118719794 Ki = 79.3 nM T67162 CG0O3Q 118719795 Ki = 42.3 nM T67162 CUHT71 118719796 Ki = 17.7 nM T67162 CR0FM7 118719797 Ki = 158 nM T67162 CPX2Y1 118719798 Ki = 94.3 nM T67162 C0KH8S 118719799 Ki = 109 nM T67162 C4YR6K 118719800 Ki = 73.5 nM T67162 CX7WL5 118719801 Ki = 46.7 nM T67162 C5TO1H 118719802 Ki = 23.7 nM T67162 CTQ71B 118719803 Ki = 272 nM T67162 C8KJ6Y 118719804 Ki = 139 nM T67162 CFL6U9 118719805 Ki = 62.7 nM T67162 CQK7O2 118719806 Ki = 162 nM T67162 CWO13F 118719807 Ki = 171 nM T67162 CZ8FE6 118719808 Ki = 62.6 nM T67162 CRH56E 118719809 Ki = 44.1 nM T67162 CUH0A6 118719810 Ki = 26.6 nM T67162 CZKW38 118719811 Ki = 12.8 nM T67162 C74DCE 118719812 Ki = 9.4 nM T67162 CT8KO4 118719925 Ki = 660.69 nM T67162 C16DHZ 118719926 Ki = 1174.9 nM T67162 CLA06I 118719927 Ki = 933.25 nM T67162 CYW82N 118721287 Ki > 1000 nM T67162 CI5MY4 118722109 IC50 > 10000 nM T67162 CES97Y 118722639 Ki = 76 nM T67162 CM3P7R 118722912 Ki > 1000 nM T67162 CP3QC2 118722913 Ki = 160 nM T67162 C1PG3C 118722914 Ki > 1000 nM T67162 CR6E5D 118722915 Ki > 1000 nM T67162 CC94IX 118725995 EC50 = 478.63 nM T67162 CL1I3E 118725996 EC50 = 112.2 nM T67162 C3AU5G 118725997 EC50 = 147.91 nM T67162 C5EVX3 118726000 EC50 = 776.25 nM T67162 CAM4W1 118726001 EC50 = 501 nM T67162 C7MVA4 118726004 EC50 > 100000 nM T67162 CP8YI2 118726005 EC50 > 100000 nM T67162 C5SIX4 118726006 EC50 = 309.03 nM T67162 C6MV1Y 118726008 EC50 > 100000 nM T67162 CH5W0A 118726009 EC50 = 389 nM T67162 CWN6M4 118726010 EC50 = 87.1 nM T67162 CM7NZ9 118726011 EC50 = 37.15 nM T67162 C8LF5G 118726014 EC50 > 100000 nM T67162 CD04WB 118726015 EC50 > 100000 nM T67162 C0OUK6 118726016 EC50 > 100000 nM T67162 CEXM41 118726017 EC50 > 100000 nM T67162 C5T1WS 118726018 EC50 > 100000 nM T67162 CK1S2U 118726021 EC50 > 100000 nM T67162 CD5RI3 118731502 Ki = 73 nM T67162 C5UQ3P 118731503 Ki = 40 nM T67162 CB6H8O 118731504 Ki = 4.8 nM T67162 CLFJ64 118731505 Ki = 14 nM T67162 CFPX32 118731506 Ki = 70 nM T67162 CL35UJ 118731507 Ki = 120 nM T67162 CF3TJ0 118731508 Ki = 31 nM T67162 CRBZ61 118731509 Ki = 160 nM T67162 CRJ4A6 118731510 Ki = 29 nM T67162 CCPL16 118731511 Ki = 62 nM T67162 C2POB0 118731512 Ki = 270 nM T67162 CZRB40 118731513 Ki = 180 nM T67162 C75OXS 118736395 Ki = 340 nM T67162 C74FCM 118736396 Ki = 68 nM T67162 C3F8PA 118736397 Ki = 215 nM T67162 COS3K9 121304408 Ki = 354.81 nM T67162 C9G3ZJ 121304414 Ki = 467.74 nM T67162 CVN57T 121304417 Ki = 537.03 nM T67162 C4RD9Y 121304424 Ki = 794.33 nM T67162 CN5YP1 121304426 Ki = 446.68 nM T67162 CJ4GF7 121304428 Ki = 39.81 nM T67162 CXL97W 121304430 Ki = 660.69 nM T67162 CA8CY5 121304437 Ki = 123.03 nM T67162 C1PKR0 121304441 Ki = 338.84 nM T67162 CQ7T4P 121304448 Ki = 426.58 nM T67162 CWLB20 121304449 Ki = 537.03 nM T67162 CC3MP6 121304452 Ki = 363.08 nM T67162 CW68KD 121304458 Ki = 676.08 nM T67162 CVA9F4 121304464 Ki = 128.82 nM T67162 CPB58L 121304467 Ki = 870.96 nM T67162 CFXN81 121304470 Ki = 309.03 nM T67162 CTCA98 121304474 Ki = 691.83 nM T67162 COB2X5 121304477 Ki = 1479.11 nM T67162 CZ0BI4 121304484 Ki = 7585.78 nM T67162 CW51NQ 121304485 Ki = 74.13 nM T67162 CX1DQ6 121304488 Ki = 954.99 nM T67162 CZ4D2Y 121304493 Ki = 1621.81 nM T67162 CU50JM 121304499 Ki = 467.74 nM T67162 C7NLV2 121304500 Ki = 691.83 nM T67162 C18GSY 121304506 Ki = 707.95 nM T67162 C21MEQ 121304510 Ki = 346.74 nM T67162 C7F3NO 121304514 Ki = 331.13 nM T67162 CPNV43 121304527 Ki = 66.07 nM T67162 CCW3A9 121304532 Ki = 891.25 nM T67162 CQ2UM4 121304538 Ki = 478.63 nM T67162 CR7L0O 121304539 Ki = 63.1 nM T67162 C2GI6S 121304542 Ki = 1230.27 nM T67162 C1AB6P 121304551 Ki = 57.54 nM T67162 CTI6Z7 121304565 Ki = 1148.15 nM T67162 CFVP28 121304568 Ki = 426.58 nM T67162 CO6JN7 121304569 Ki = 501.19 nM T67162 CN05ZQ 121304574 Ki = 1862.09 nM T67162 CU0M7B 121304590 Ki = 660.69 nM T67162 C3FPD2 121304592 Ki = 3801.89 nM T67162 C73GOE 121304594 Ki = 977.24 nM T67162 CLZK90 121304596 Ki = 1548.82 nM T67162 C6YLM8 121304597 Ki = 389.05 nM T67162 CX5MO3 121304598 Ki = 457.09 nM T67162 C12GJP 121304609 Ki = 1288.25 nM T67162 C6DT8C 121304616 Ki = 537.03 nM T67162 CZS7C4 121304618 Ki = 2187.76 nM T67162 CDQ35E 121304633 Ki = 794.33 nM T67162 C31AEQ 121304649 Ki = 25.7 nM T67162 C9TYS1 121304653 Ki = 295.12 nM T67162 C2VTK5 121304654 Ki = 1148.15 nM T67162 CSYD40 121304673 Ki = 512.86 nM T67162 C6IB0P 121304685 Ki = 1348.96 nM T67162 CU0L6A 121304697 Ki = 933.25 nM T67162 CNOW27 121304705 Ki = 851.14 nM T67162 C6NA0P 121304710 Ki = 524.81 nM T67162 CXC70Q 121304711 Ki = 724.44 nM T67162 CE0ND7 121304744 Ki = 218.78 nM T67162 C1MZ6T 121304754 Ki = 1698.24 nM T67162 CU93LN 121304777 Ki = 954.99 nM T67162 C5HQ4S 121304867 Ki = 165.96 nM T67162 CAS0Y9 121315197 Ki = 977.24 nM T67162 CG92LO 121315203 Ki = 436.52 nM T67162 CRZ1V0 121315205 Ki = 61.66 nM T67162 CV3XH6 121315206 Ki = 123.03 nM T67162 C4TI7P 121315244 Ki = 107.15 nM T67162 CLM9E8 121315259 Ki = 501.19 nM T67162 C7B3XN 121315293 Ki = 512.86 nM T67162 C9U5CV 121315295 Ki = 794.33 nM T67162 C6UMN2 121315304 Ki = 1584.89 nM T67162 CH5FS4 121315329 Ki = 1778.28 nM T67162 CX71KH 121315331 Ki = 3311.31 nM T67162 CV4EO5 121315336 Ki = 478.63 nM T67162 CN39AK 121315339 Ki = 616.6 nM T67162 CFWG90 121315351 Ki = 467.74 nM T67162 C14NCL 121315356 Ki = 295.12 nM T67162 COG90M 121315374 Ki = 501.19 nM T67162 CEY62R 121315401 Ki = 162.18 nM T67162 C0NB3Y 121315426 Ki = 1380.38 nM T67162 C0E6HD 121315586 Ki = 66.07 nM T67162 CA7HL6 121315615 Ki = 1348.96 nM T67162 CBAG84 121315634 Ki = 331.13 nM T67162 C3YT2R 121418441 EC50 = 120 nM T67162 CVS9K7 121418491 EC50 = 61 nM T67162 C5OC0E 121418538 EC50 = 10 nM T67162 C35WTP 122177641 Ki = 1.6 nM T67162 C8OS7B 122177642 Ki = 4.9 nM T67162 CV2AT4 122177644 Ki = 18 nM T67162 CB16GY 122177645 Ki = 0.47 nM T67162 C5TI4H 122179561 EC50 = 218.78 nM T67162 C14PNH 122179562 EC50 = 1413 nM T67162 C6VI4R 122179563 EC50 = 41.69 nM T67162 C03ORH 122179564 EC50 = 4677 nM T67162 CP6VX4 122180568 Ki = 31.5 nM T67162 CU0L3S 122180569 Ki = 57.2 nM T67162 C87MAH 122180570 Ki = 51.8 nM T67162 CY9BN0 122180571 Ki = 83.4 nM T67162 CS9NY8 122180572 Ki = 80.8 nM T67162 CAL57I 122180573 Ki = 424 nM T67162 CZ72GE 122180574 Ki = 46.6 nM T67162 CZ4M2F 122180575 Ki = 23.3 nM T67162 C03CGT 122180576 Ki = 50.1 nM T67162 C2X3ZW 122180610 Ki = 43.7 nM T67162 CRMS80 122180611 Ki = 42.5 nM T67162 CWO2Y4 122180612 Ki = 69 nM T67162 C2DZ0K 122180613 Ki = 103 nM T67162 CH81IV 122180614 Ki = 885 nM T67162 C1EPB8 122180615 Ki = 56.1 nM T67162 CV26IM 122180616 Ki = 53.9 nM T67162 CQ0L6Z 122180617 Ki = 2590 nM T67162 CVX5Y3 122180618 Ki = 189 nM T67162 CEGV53 122180619 Ki = 819 nM T67162 CV1OA4 122180620 Ki = 1210 nM T67162 CYID81 122180621 Ki = 1020 nM T67162 CB91ZG 122180622 Ki = 607 nM T67162 C1CIH2 122180623 Ki = 424 nM T67162 C8YZ9Q 122180624 Ki = 18800 nM T67162 C9S3VH 122180625 Ki = 15100 nM T67162 CQ3N6G 122180626 Ki = 789 nM T67162 C6YL5S 122180627 Ki = 963 nM T67162 CPRB82 122180954 Ki = 4 nM T67162 C08BVN 122180955 Ki = 3.9 nM T67162 CH9SX5 122180956 Ki = 73 nM T67162 CAJ9N8 122181005 Ki = 244 nM T67162 C90VEH 122181006 Ki = 268 nM T67162 CN7TP8 122181007 Ki = 54.7 nM T67162 CCV9D5 122181326 Ki = 34 nM T67162 C91LDR 122181327 Ki = 7.5 nM T67162 CPW19F 122181328 Ki = 6.6 nM T67162 C5D1NC 122181329 Ki = 2.9 nM T67162 C05RGV 122181330 Ki = 23 nM T67162 C1KWI9 122181331 Ki = 13 nM T67162 CQ35XD 122181332 Ki = 12 nM T67162 C3XGN0 122181333 Ki = 13 nM T67162 C3BTQ7 122181334 Ki = 46.9 nM T67162 CXL5V3 122183764 EC50 = 200 nM T67162 CK3VT8 122183765 Ki = 43.1 nM T67162 CQ6CW2 122183766 Ki = 885 nM T67162 CQE64Y 122183767 Ki = 39.2 nM T67162 CI43NJ 122183768 Ki = 827 nM T67162 CK6D3O 122183769 Ki = 53 nM T67162 CC2WO0 122183770 Ki = 72.3 nM T67162 C12TRH 122183771 Ki = 12.9 nM T67162 CZO5G4 122183772 Ki = 13.8 nM T67162 C8V5TM 122183773 Ki = 14.8 nM T67162 CH4J7G 122183774 Ki = 8.37 nM T67162 CKIP60 122183775 Ki = 929 nM T67162 C8AK5V 122183776 Ki = 68.2 nM T67162 CS65WU 122183777 Ki = 1000 nM T67162 C06GQO 122183778 Ki = 915 nM T67162 C8YL2R 122183779 Ki = 34.1 nM T67162 CQ4YF9 122183780 Ki = 682 nM T67162 C7ZNJ8 122183781 Ki = 707 nM T67162 C4U8LC 122183782 Ki = 774 nM T67162 CLA65S 122183783 Ki = 1030 nM T67162 CIG04A 122186385 Ki = 5586 nM T67162 C6UI5G 122186390 Ki = 175 nM T67162 C6LN7X 122186408 Ki = 197 nM T67162 CK5BP3 122189387 Ki = 81 nM T67162 C8JV3W 122189388 Ki = 3.8 nM T67162 CV1U4Q 122189389 Ki = 51 nM T67162 C4PBA3 122189390 Ki = 8 nM T67162 CD7UN3 122189391 Ki = 9.4 nM T67162 C14FCX 122189392 Ki = 10 nM T67162 C1NIK8 122189393 Ki = 54 nM T67162 C9KXH4 122189394 Ki = 7.3 nM T67162 C87LIY 122191600 Ki = 7500 nM T67162 CPF1G4 122191601 Ki = 920 nM T67162 C3ZR7F 122191602 Ki = 520 nM T67162 CI5L4E 122191603 Ki = 220 nM T67162 C9AH4E 122191604 Ki = 430 nM T67162 CVJ3R4 122191605 Ki = 48 nM T67162 CSR76G 122191606 Ki = 120 nM T67162 C2J4ZX 122191607 Ki = 51 nM T67162 CM84TD 122191608 Ki = 4000 nM T67162 C94XIT 122191609 Ki = 5200 nM T67162 C7UVD4 122191610 Ki = 4100 nM T67162 CWH1P8 122191611 Ki = 920 nM T67162 C71KZQ 122205437 Ki = 45 nM T67162 C30ZRC 122205438 Ki = 1.5 nM T67162 CBHT01 122377930 Ki = 102 nM T67162 C6TEJ0 126532768 Ki = 251.19 nM T67162 CNRI41 126533424 Ki = 316.23 nM T67162 CG65RM 126533453 Ki = 316.23 nM T67162 CRX67M 126533461 Ki = 199.53 nM T67162 C0OPY6 126533669 Ki = 251.19 nM T67162 CSN21X 126533798 Ki = 199.53 nM T67162 CMHY08 126533799 Ki = 398.11 nM T67162 CP8W0X 126533801 Ki = 251.19 nM T67162 CXM45K 126533810 Ki = 158.49 nM T67162 C0E7OY 126533847 Ki = 630.96 nM T67162 CPL62Z 126533872 Ki = 31.62 nM T67162 C1ST0Y 126533877 Ki = 398.11 nM T67162 CDP5C4 126533939 Ki = 199.53 nM T67162 CX2A4N 126533957 Ki = 630.96 nM T67162 CIV7R0 126533969 Ki = 199.53 nM T67162 CC7V5Y 126533978 Ki = 19.95 nM T67162 CI97TU 126533981 Ki = 158.49 nM T67162 CON63X 126534012 Ki = 158.49 nM T67162 C9G1IV 126534022 Ki = 39.81 nM T67162 C9AN4B 126534041 Ki = 398.11 nM T67162 C8JKG0 126534069 Ki = 794.33 nM T67162 CA4QM3 126534084 Ki = 251.19 nM T67162 C3SUR8 126534086 Ki = 251.19 nM T67162 CCX0O5 126534178 Ki = 630.96 nM T67162 C6NU0Y 126534182 Ki = 6309.57 nM T67162 CNUA81 126534195 Ki = 158.49 nM T67162 CIAD86 126534204 Ki = 630.96 nM T67162 C4R7XU 126534291 Ki = 398.11 nM T67162 CVBX50 126534373 Ki = 50.12 nM T67162 CB94HO 126534441 Ki = 398.11 nM T67162 CSX9W5 126534443 Ki = 1584.89 nM T67162 CQ39ZD 126534462 Ki = 199.53 nM T67162 CT75WF 126534466 Ki = 316.23 nM T67162 C52IHK 126534498 Ki = 501.19 nM T67162 CFA3D6 126534516 Ki = 125.89 nM T67162 CX14VB 126534676 Ki = 31.62 nM T67162 CIW18V 126534678 Ki = 100 nM T67162 CJPA49 126534738 Ki = 158.49 nM T67162 CG7CY3 126534740 Ki = 31.62 nM T67162 CQDE96 126534746 Ki = 316.23 nM T67162 CIN62J 126534758 Ki = 100 nM T67162 CXI58O 126534764 Ki = 316.23 nM T67162 C0WUJ5 126534771 Ki = 158.49 nM T67162 CFDR90 126534824 Ki = 1258.93 nM T67162 CX9LM7 126534859 Ki = 1000 nM T67162 CKN57U 126534860 Ki = 398.11 nM T67162 C3YB2Z 126534863 Ki = 158.49 nM T67162 CR70LT 126534933 Ki = 501.19 nM T67162 CKBT37 126534948 Ki = 501.19 nM T67162 C6DLR7 126534986 Ki = 316.23 nM T67162 CR10PO 126534991 Ki = 1258.93 nM T67162 CFT24J 126535001 Ki = 100 nM T67162 C58EIM 126535029 Ki = 630.96 nM T67162 C5HQB6 126535034 Ki = 10 nM T67162 C9Q0VB 126535075 Ki = 501.19 nM T67162 CMT3Q8 126535410 Ki = 398.11 nM T67162 C5YS6F 126535470 Ki = 630.96 nM T67162 C4TZ6I 126535517 Ki = 630.96 nM T67162 CM57GR 126720252 Ki = 8210 nM T67162 CLWM12 126720394 Ki = 6100 nM T67162 C8Q1JB 126720403 Ki = 3436 nM T67162 C1U3SZ 126720425 Ki = 2941 nM T67162 C5G8FD 126720440 Ki = 3482 nM T67162 CCF0J2 127024958 Ki = 5031 nM T67162 C82TLX 127024959 Ki = 310 nM T67162 C2MWE6 127024960 Ki = 12143 nM T67162 CIHZ54 127025242 Ki = 199 nM T67162 CCY7P3 127025243 Ki = 60 nM T67162 C9AQH0 127025258 Ki = 302 nM T67162 CH1CG6 127025275 Ki = 911 nM T67162 CG3N7S 127025276 Ki = 13 nM T67162 CGO8I5 127025277 Ki = 482 nM T67162 CJZC96 127025278 Ki = 322 nM T67162 CTBN56 127026052 Ki = 2454.71 nM T67162 CG8Q4L 127026123 Ki = 404 nM T67162 CTYP30 127026133 Ki = 94 nM T67162 CX6EI2 127026750 Ki = 322 nM T67162 C2YDB4 127027076 Ki = 1553 nM T67162 CU59DP 127027077 Ki = 373 nM T67162 CI94GN 127027078 Ki = 95 nM T67162 C2H6GE 127027079 Ki = 52 nM T67162 C5G4AH 127027080 Ki = 131 nM T67162 C9PNV3 127027384 Ki = 55 nM T67162 C09YOS 127027905 Ki > 10000 nM T67162 CH2BP0 127027974 Ki = 1549 nM T67162 CXQ94C 127028034 Ki = 34 nM T67162 CY2TW9 127028152 Ki = 2906 nM T67162 CAZJ04 127028153 Ki = 5187 nM T67162 CR48GO 127028154 Ki = 1709 nM T67162 CE9MN1 127028185 Ki > 10000 nM T67162 C8MC1I 127028408 Ki = 4897.79 nM T67162 CD8H7W 127028471 Ki = 839 nM T67162 C4EAY5 127028472 Ki = 127 nM T67162 CUS8R9 127028473 Ki = 931 nM T67162 C9SC6E 127028505 Ki > 10000 nM T67162 CZ26YR 127028797 Ki = 302 nM T67162 CI2R1N 127028798 Ki = 1814 nM T67162 CS8GJ5 127028799 Ki = 5641 nM T67162 CU0WQ3 127029375 Ki = 4255 nM T67162 CS1GX5 127029649 Ki = 6790 nM T67162 C9N3BE 127029650 Ki = 1976 nM T67162 CQFS48 127029651 Ki = 2261 nM T67162 C7F3YE 127029652 Ki = 261 nM T67162 C1RF0I 127031156 Ki = 3162.28 nM T67162 CJ4YC0 127031397 Ki = 283 nM T67162 CE1IA7 127031399 Ki = 211 nM T67162 C4WKG9 127031403 Ki = 54 nM T67162 CEDM28 127031404 Ki = 1095 nM T67162 CV5UH0 127031405 Ki > 10000 nM T67162 CHN9X2 127031422 Ki = 159 nM T67162 C0CY9W 127031423 Ki = 99 nM T67162 CNH2V8 127031424 Ki = 121 nM T67162 C0A3PY 127031458 Ki = 6309.57 nM T67162 C2W0HL 127031949 Ki > 10000 nM T67162 CZ61LK 127034966 EC50 > 5011.87 nM T67162 CA0SN5 127034967 EC50 > 5011.87 nM T67162 CQ0ZT9 127035062 Ki = 1729 nM T67162 CO53TS 127035828 Ki > 1000 nM T67162 CY7LP9 127035829 Ki > 1000 nM T67162 CR29BS 127035830 Ki > 1000 nM T67162 CU49VE 127036186 Ki = 5128.61 nM T67162 CG06BD 127036932 Ki = 1862.09 nM T67162 CVW71O 127036953 Ki = 4365.16 nM T67162 C7N5DF 127037679 Ki = 147 nM T67162 CTE43C 127037681 Ki = 140 nM T67162 CT1Z3P 127037852 Ki = 10000 nM T67162 CH6KI9 127037866 Ki = 10000 nM T67162 C2XBE8 127037921 Ki = 230 nM T67162 CX0CN4 127037922 Ki = 37 nM T67162 CDAE15 127038033 Ki = 104 nM T67162 C81TYN 127038069 Ki = 6230 nM T67162 C0SWK3 127038076 Ki = 1290 nM T67162 C3QL9U 127038078 Ki = 79630 nM T67162 C8TC9G 127038281 Ki = 16 nM T67162 CP8T3I 127039208 Ki = 15848.93 nM T67162 CYJ2D5 127039593 Ki = 18 nM T67162 CBF6T8 127039745 EC50 = 3.23 nM T67162 CLY0X5 127039746 EC50 = 32.7 nM T67162 CES26L 127039755 Ki = 85 nM T67162 CAW01Z 127040356 Ki = 12589.25 nM T67162 CZ6V5D 127040357 Ki > 10000 nM T67162 CE95PL 127040381 Ki = 6309.57 nM T67162 C37KDY 127040382 Ki > 10000 nM T67162 CX1W5M 127040442 Ki = 51 nM T67162 C6Z9VL 127040695 Ki = 25118.86 nM T67162 CQGJ12 127040696 Ki = 7943.28 nM T67162 CWC31L 127040697 Ki = 12589.25 nM T67162 CF31EG 127040698 Ki = 15848.93 nM T67162 CMH9E6 127040712 Ki = 10000 nM T67162 CG74QA 127040713 Ki = 25118.86 nM T67162 CZ58KA 127040714 Ki = 15848.93 nM T67162 C34BGK 127040715 Ki = 10000 nM T67162 CL4WG3 127040716 Ki = 15848.93 nM T67162 C8D4AV 127040908 Ki = 50 nM T67162 C53WRO 127041026 Ki = 19952.62 nM T67162 C15BGV 127041244 Ki = 60 nM T67162 CU0J4S 127041258 Ki = 45 nM T67162 C20MZH 127041259 Ki = 46 nM T67162 CP16CZ 127041260 Ki = 360 nM T67162 CZT53S 127041261 Ki = 290 nM T67162 C0S5MT 127041332 Ki > 31622.78 nM T67162 C5B1AG 127041347 Ki = 15848.93 nM T67162 C0J8HC 127041348 Ki = 1584.89 nM T67162 C8MG6H 127041349 Ki = 10000 nM T67162 C87MZF 127041350 Ki = 7943.28 nM T67162 C0FJP2 127041563 Ki = 324 nM T67162 CUC3F9 127041564 Ki = 280 nM T67162 C9D7SK 127041673 Ki = 7943.28 nM T67162 COG9D2 127041874 Ki = 52 nM T67162 CS78AZ 127041951 Ki > 10000 nM T67162 CU9C4S 127041952 Ki = 12589.25 nM T67162 C9HPT6 127041953 Ki > 10000 nM T67162 CS4WH1 127042184 Ki = 54 nM T67162 C13AIN 127042185 Ki = 35 nM T67162 C4FG7S 127042371 EC50 = 21.6 nM T67162 C7ETU0 127042372 EC50 = 39.4 nM T67162 CR59TP 127042539 Ki = 15 nM T67162 C54IZC 127042540 Ki = 20 nM T67162 C8G1HF 127042841 Ki = 160 nM T67162 C83YZJ 127045665 Ki > 2000 nM T67162 CM02RK 127045814 Ki = 13.2 nM T67162 C35GAL 127045853 Ki = 65 nM T67162 C17LBT 127045854 EC50 = 7.3 nM T67162 CJ8GS7 127045855 EC50 = 170 nM T67162 C9EH4D 127045870 Ki > 2000 nM T67162 C9CRG7 127045871 Ki = 640 nM T67162 C06KDX 127045872 Ki > 2000 nM T67162 CRYE28 127045873 Ki = 1231 nM T67162 CX84AD 127045874 Ki = 25 nM T67162 CT15OK 127046255 Ki = 8.08 nM T67162 C3WNA8 127046749 Ki = 5120 nM T67162 C4Q6DY 127046815 Ki = 86 nM T67162 CF4X5D 127046817 Ki = 205 nM T67162 CZU72I 127046818 Ki > 2000 nM T67162 CF4E8W 127046819 Ki = 382 nM T67162 C59QDV 127046922 EC50 = 0.3 nM T67162 C2E1ZA 127046948 Ki = 2300 nM T67162 CTI5Z8 127046949 EC50 = 17 nM T67162 C4D6BQ 127046950 Ki = 67 nM T67162 CM4CQ7 127046951 Ki = 1700 nM T67162 C29ERQ 127046952 Ki = 63 nM T67162 C38UBC 127046963 Ki > 2000 nM T67162 CH6W2T 127046982 Ki = 367 nM T67162 C9DFA6 127047182 EC50 = 5300 nM T67162 C78IFA 127047221 Ki = 200 nM T67162 CFOD25 127047227 Ki = 12.8 nM T67162 C5CG1O 127047229 EC50 = 0.9 nM T67162 CN3B7M 127047230 Ki = 15.5 nM T67162 CU2ST0 127047318 EC50 = 2600 nM T67162 C6TMB2 127047319 EC50 = 37.6 nM T67162 CB80KL 127047458 EC50 = 4100 nM T67162 C1D7PX 127047462 EC50 = 3500 nM T67162 C84PLD 127047536 Ki > 2000 nM T67162 C17RWQ 127047537 Ki > 2000 nM T67162 C7OCX9 127047538 Ki = 52 nM T67162 C0RE8Z 127047592 EC50 = 14000 nM T67162 C71MFW 127047640 EC50 > 10000 nM T67162 C6P4OZ 127047641 EC50 = 9900 nM T67162 CJH46E 127047680 Ki = 1700 nM T67162 CUC1G6 127047776 Ki = 547 nM T67162 CZL0U7 127047859 EC50 = 2.6 nM T67162 C4SG7L 127047870 Ki = 12.5 nM T67162 CV1KL4 127047898 Ki = 614 nM T67162 C3BU0X 127047899 Ki = 630 nM T67162 C7W4MF 127047900 Ki = 113 nM T67162 CLK3C5 127047901 Ki = 22 nM T67162 CZ6XL5 127047996 EC50 = 25 nM T67162 C3G8BQ 127048020 Ki = 5.47 nM T67162 C0V5YU 127048532 IC50 = 1580 nM T67162 CHW0L2 127048533 IC50 = 202 nM T67162 C9QR6V 127048539 IC50 = 43 nM T67162 CU6K4P 127048540 IC50 = 30 nM T67162 CC7BU0 127049059 Ki = 10 nM T67162 C42FHY 127049060 Ki = 22 nM T67162 CF2QY9 127049061 Ki = 213.8 nM T67162 CN2F1W 127049163 IC50 = 4.1 nM T67162 C1TI6J 127049515 IC50 = 39.4 nM T67162 CT16PL 127049516 IC50 = 3600 nM T67162 C4QKS3 127049517 IC50 = 12 nM T67162 C03BLH 127049522 IC50 = 167 nM T67162 C2IX7Q 127049847 IC50 = 34.9 nM T67162 CRK8W3 127049848 IC50 = 89.8 nM T67162 C85PIF 127049849 IC50 = 37.7 nM T67162 CO2V5Z 127049850 IC50 = 58.5 nM T67162 C27MWC 127049861 IC50 = 70 nM T67162 CZS1L6 127049862 IC50 = 8.5 nM T67162 CZD91J 127049863 IC50 = 23 nM T67162 C1S6EN 127049864 IC50 = 10 nM T67162 C2H0BQ 127049865 IC50 = 12 nM T67162 CUK1S9 127049866 IC50 = 91 nM T67162 CX53AC 127050632 Ki = 18 nM T67162 CP9UT4 127050764 IC50 = 98.4 nM T67162 C9T2VY 127050765 IC50 = 32 nM T67162 CIOZ65 127051038 IC50 = 55 nM T67162 C7XK3G 127051039 IC50 = 116 nM T67162 CR4TV6 127051040 IC50 = 16.8 nM T67162 CCTO35 127051041 IC50 = 9.8 nM T67162 CA2SJ6 127051340 IC50 = 171 nM T67162 CTL0S1 127051516 Ki = 23.99 nM T67162 CTL8J1 127051843 Ki = 1445.44 nM T67162 CF6V9Q 127051844 Ki = 218 nM T67162 C8TNB1 127051845 Ki = 249 nM T67162 CT9O7G 127051863 Ki = 438 nM T67162 C5ONG1 127051864 Ki = 44 nM T67162 CVQW26 127051865 Ki = 180 nM T67162 CRF85X 127052458 Ki = 363.08 nM T67162 CCY71I 127052465 Ki > 10000 nM T67162 C2E9VX 127052467 Ki = 158.49 nM T67162 CPO4C3 127052468 Ki = 1150 nM T67162 CSQ2N8 127052486 Ki = 95 nM T67162 C4YJ8H 127052487 Ki = 134 nM T67162 CT9RS4 127052488 Ki = 194.98 nM T67162 CLU7C1 127052757 Ki = 316.23 nM T67162 C95KYT 127052758 Ki = 165.96 nM T67162 CYNR02 127052759 Ki = 123 nM T67162 C14YJU 127052778 Ki = 158.49 nM T67162 C1JAS7 127052779 Ki = 758.58 nM T67162 C7MQK8 127053042 Ki = 422 nM T67162 C3WIA6 129103318 IC50 = 9.02 nM T67162 CBX2V6 129186527 IC50 = 31.5 nM T67162 CV2K7I 129186528 IC50 = 5.49 nM T67162 CD9C1F 129186530 IC50 = 6660 nM T67162 C2F5YE 129186531 IC50 = 5530 nM T67162 C6GC0F 129186534 IC50 = 3.32 nM T67162 CTP0O3 129186549 IC50 = 75.4 nM T67162 C8KM6N 129186554 IC50 = 2.61 nM T67162 C7FR6U 129186558 IC50 = 960 nM T67162 CEZT92 129186564 IC50 = 3.51 nM T67162 C10VDB 130431277 Ki = 139 nM T67162 CI1NF8 130431279 Ki = 619 nM T67162 CS8O4E 130431287 Ki = 137 nM T67162 C75AQS 130431288 Ki = 891 nM T67162 C85MOW 130431289 Ki = 247 nM T67162 CR7T6X 130431290 Ki = 12.5 nM T67162 C2OH7B 130431291 Ki = 10800 nM T67162 C2AZ0H 130431294 Ki = 21400 nM T67162 CEQ43Y 130431295 Ki = 20800 nM T67162 CK64GU 130431296 Ki = 328 nM T67162 CU9XL0 130431303 Ki = 150 nM T67162 CB6Q3Y 130431306 Ki = 18900 nM T67162 C3MA6H 130431309 Ki = 193 nM T67162 CYW0X2 130431314 Ki = 75.8 nM T67162 C8ZED9 130431315 Ki = 80.2 nM T67162 CDN26V 130431316 Ki = 132 nM T67162 CL64UW 130431317 Ki = 164 nM T67162 C8HE2O 130431318 Ki = 11400 nM T67162 CZ6S4T 130431319 Ki = 219 nM T67162 C8ZHI7 130431325 Ki = 6.34 nM T67162 CF5SW8 130431328 Ki = 13500 nM T67162 CN9RZ3 130431329 Ki = 10800 nM T67162 CEP1Q6 130431334 Ki = 6.83 nM T67162 CWT8I6 130431336 Ki = 16.1 nM T67162 CN70MW 130431337 Ki = 5.5 nM T67162 CIXV41 130431340 Ki = 12.2 nM T67162 C4GF1U 130431342 Ki = 1620 nM T67162 CWAC20 130431343 Ki = 5.64 nM T67162 C2WI5R 130431351 Ki = 27.8 nM T67162 C50GOC 130442480 Ki = 9600 nM T67162 CM04RF 130442572 Ki = 7600 nM T67162 CLP6B7 130816094 Ki = 2340 nM T67162 C52QWM 131801150 EC50 = 2.9 nM T67162 CTVU23 131801153 EC50 = 0.71 nM T67162 CZBL63 131801154 EC50 = 6.3 nM T67162 C3HI8S 132141090 Ki = 630.96 nM T67162 CU5F7W 132141173 Ki = 1445.44 nM T67162 C5P9AV 132153537 Ki = 870.96 nM T67162 C3CVU2 132156264 Ki = 2570.4 nM T67162 C9W4AK 132156266 Ki = 1230.27 nM T67162 CRH07J 132156331 Ki = 117.49 nM T67162 CF5V3G 132156412 Ki = 630.96 nM T67162 CCL8F6 132495282 Ki > 10000 nM T67162 C4LJ2Y 132503215 Ki = 36 nM T67162 CM8B1L 132525569 Ki = 466 nM T67162 CU5L0K 132525570 Ki = 37 nM T67162 CVZ57M 132578416 EC50 = 0.27 nM T67162 CAVB41 132584404 Ki > 10000 nM T67162 CY4CU6 132606870 Ki = 182 nM T67162 CVYX78 132606872 Ki = 695 nM T67162 CS0MB3 132938109 Ki = 343 nM T67162 C6Z5UG 134129927 Ki = 794.33 nM T67162 CLW62U 134131970 Ki = 251.19 nM T67162 C0RQC6 134131976 Ki = 1385 nM T67162 C7UOA9 134132432 Ki > 10000 nM T67162 CQX4U3 134133064 Ki = 2933 nM T67162 CCPI30 134133464 Ki = 0.72 nM T67162 CTS3J4 134133483 Ki = 260 nM T67162 C0J2ML 134133604 Ki = 946 nM T67162 CM0TS6 134133967 Ki = 269.15 nM T67162 CR8HL3 134134147 Ki = 1445.44 nM T67162 CC1DO8 134134456 Ki = 522 nM T67162 CR4F6X 134135492 Ki = 18 nM T67162 CM34TY 134135507 Ki = 9.6 nM T67162 C2Q3JY 134135516 Ki = 537 nM T67162 CJ6C3E 134135947 Ki = 107 nM T67162 CJG3U0 134136134 Ki = 64 nM T67162 CFOU70 134136921 Ki = 15848.93 nM T67162 C87ZJW 134137152 Ki > 10000 nM T67162 CSM98N 134137323 Ki = 331 nM T67162 C08ZBY 134137332 Ki = 393 nM T67162 CD41CW 134137432 Ki = 0.3 nM T67162 CXF52V 134137560 Ki = 177 nM T67162 CN4LI8 134137732 Ki = 295 nM T67162 C50WSG 134137966 Ki = 1995.26 nM T67162 C90XZH 134138881 Ki = 2.1 nM T67162 CTP83K 134139510 Ki = 1.9 nM T67162 CRC2V0 134139826 Ki = 685 nM T67162 CHK39T 134141166 Ki = 293 nM T67162 CLW86T 134141354 Ki = 3548.13 nM T67162 CXC80B 134142146 Ki = 10 nM T67162 C6PSI9 134142907 Ki = 4346 nM T67162 CVJ70S 134143778 Ki = 0.85 nM T67162 CJE86B 134143833 Ki = 41 nM T67162 CL8I1U 134144243 Ki = 1737.8 nM T67162 CR5L4K 134144303 Ki = 1170 nM T67162 C80TGJ 134144864 Ki = 375 nM T67162 CK5RU9 134145903 Ki = 53 nM T67162 C8AZ1F 134146083 Ki = 14 nM T67162 C8RI0E 134146106 Ki = 15 nM T67162 C2E0ID 134146185 Ki = 2766 nM T67162 CC9P2T 134146194 Ki = 1087 nM T67162 CZDH24 134147097 Ki = 1000 nM T67162 CV0QZ5 134147124 Ki = 268 nM T67162 CB0NS6 134147903 Ki = 23 nM T67162 C41XSD 134147935 Ki = 1959 nM T67162 CH21YW 134148634 Ki > 10000 nM T67162 CJ5W4V 134149077 Ki = 104 nM T67162 CBU81N 134149168 Ki > 10000 nM T67162 CSE17M 134150535 Ki = 6309.57 nM T67162 C0S2VH 134150637 Ki = 1000 nM T67162 C5DX6R 134150645 Ki = 731 nM T67162 C6NYU2 134150754 Ki = 338.84 nM T67162 C2MAK7 134150852 Ki = 398 nM T67162 C6O8QW 134150900 Ki = 15848.93 nM T67162 CE6LN3 134151118 Ki = 75 nM T67162 CLU34D 134151427 Ki = 2583.5 nM T67162 C2JN8Y 134151729 Ki = 243 nM T67162 C8BI7V 134151764 Ki = 70 nM T67162 CK23XB 134151891 Ki = 2.8 nM T67162 CNC39L 134151926 Ki > 10000 nM T67162 C76BZW 134151980 Ki = 136 nM T67162 CIV4H5 134152583 Ki = 3460 nM T67162 CI0G7H 134153418 Ki = 26 nM T67162 CB6M5Y 134153538 Ki = 851.14 nM T67162 C42ZDI 134153624 Ki > 10000 nM T67162 CX4W7F 134153716 Ki = 243 nM T67162 C79TEI 134154068 Ki = 138 nM T67162 C9DQ4Y 134154208 Ki = 0.51 nM T67162 CMJ1U3 134154387 Ki = 5623.41 nM T67162 C4VGJ5 134154679 Ki = 416.87 nM T67162 CU6C4G 134154943 Ki = 8.9 nM T67162 C6QAY2 134155116 Ki = 750 nM T67162 C79QLN 134155460 Ki = 812.83 nM T67162 CIUZ94 134155476 Ki = 116 nM T67162 C90QNV 134155645 Ki = 178 nM T67162 C0AE1P 134156091 Ki = 2511.89 nM T67162 CVR87Q 134156222 Ki = 5370.32 nM T67162 CAB4K6 134156305 Ki = 308 nM T67162 C50XNE 134156520 Ki = 36 nM T67162 CUHE07 134157171 Ki = 321 nM T67162 C08MHZ 134157446 Ki = 18 nM T67162 CL6DN0 134157769 Ki = 419 nM T67162 C1GY2T 135156251 EC50 > 10000 nM T67162 CRI9X8 135404757 Ki = 1099 nM T67162 C5OU1T 135409492 Ki = 119 nM T67162 C4DZ5M 135418440 Ki > 4000 nM T67162 CI4U9T 135442113 Ki = 183 nM T67162 CQ0SY6 135458464 Ki = 3.4 nM T67162 CZXW36 135469096 Ki > 4000 nM T67162 CINW45 135471592 Ki = 183 nM T67162 C8XYU4 135481864 Ki = 2011 nM T67162 C1MTS9 135492584 Ki = 2540 nM T67162 C3Q8AT 135501649 Ki = 2596 nM T67162 C7RQ2Y 135506137 Ki > 4000 nM T67162 C0TY5Z 135514603 IC50 = 30 nM T67162 C4PM9W 135515431 Ki = 22 nM T67162 C2U1EP 135524323 Ki = 130 nM T67162 CNI90F 135797785 Ki > 2000 nM T67162 CNQ47X 135846033 Ki = 1000 nM T67162 CE40DG 135882460 Ki = 7881 nM T67162 CG95BM 135887931 Ki = 2745 nM T67162 CQYI85 135887934 Ki = 543 nM T67162 C5W7CT 135887940 Ki = 280 nM T67162 C9Z6HJ 135921193 Ki = 280 nM T67162 C5KE3N 135986088 Ki = 285 nM T67162 CJEK87 135995891 Ki = 4400 nM T67162 CCP6D9 136020061 Ki = 3.162 nM T67162 CKJ02O 136020062 IC50 = 1096.48 nM T67162 C3VZ0H 136020063 IC50 = 11000 nM T67162 CH3FL1 136020067 Ki = 245.47 nM T67162 CG6KZ0 136020068 IC50 > 10000 nM T67162 CE06AS 136020090 Ki = 8.913 nM T67162 C4GLA0 136043854 Ki = 29 nM T67162 CS7ZU5 136043855 Ki = 8 nM T67162 CQC47B 136043856 Ki = 177 nM T67162 CF2BK1 136043857 Ki = 80 nM T67162 CP3XN7 136043859 Ki = 65 nM T67162 C89VLZ 136056636 Ki = 2.3 nM T67162 CZR53O 136072267 Ki = 94 nM T67162 CR3GK4 136079154 Ki = 1.349 nM T67162 CYUQ94 136079159 Ki = 1.23 nM T67162 CCEF36 136094866 Ki = 149 nM T67162 C96ZXY 136094867 Ki = 136 nM T67162 CUG28I 136117980 Ki > 2000 nM T67162 CWP0V5 136216703 Ki = 3200 nM T67162 CKJY95 137040409 Ki = 398.11 nM T67162 CA18HL 137210067 Ki = 108 nM T67162 C9EIP8 137631570 IC50 = 157 nM T67162 CA9L5S 137631807 EC50 = 53.8 nM T67162 CHM36P 137631892 Ki = 121 nM T67162 C1VMC5 137631956 Ki = 1440 nM T67162 C5QI2K 137632035 Ki = 18.5 nM T67162 C3LDV7 137632586 Ki = 1500 nM T67162 CN8BJ2 137632607 Ki = 56 nM T67162 C3R2LO 137632761 Ki = 0.54 nM T67162 C3PF9Z 137633454 Ki = 200 nM T67162 CSA30N 137633662 Ki = 14.4 nM T67162 COF9I6 137633705 Ki = 0.5 nM T67162 CU01TV 137633827 Ki = 4287 nM T67162 C8YM6U 137633863 EC50 = 0.4365 nM T67162 CN1I7A 137634153 Ki = 6000 nM T67162 C6FRJ5 137634397 Ki = 0.67 nM T67162 CM54XV 137635157 EC50 = 24.6 nM T67162 CC51JN 137635185 Ki = 4351 nM T67162 CNR82A 137635294 IC50 = 5.2 nM T67162 CPHI76 137635364 Ki = 21 nM T67162 C6DH9X 137635433 IC50 = 2.4 nM T67162 C8ZFQ6 137635685 Ki = 25 nM T67162 C0K3AP 137635725 IC50 = 6.2 nM T67162 C6QB9W 137635734 Ki = 5754.4 nM T67162 CGEQ16 137635743 Ki = 1400 nM T67162 C94VXJ 137635884 Ki = 17 nM T67162 C05XCQ 137635978 Ki = 3.2 nM T67162 CZ36LE 137636066 Ki = 1.6 nM T67162 CIV34M 137636185 Ki = 8300 nM T67162 CAL1W4 137636298 Ki = 1200 nM T67162 CX8O0V 137636308 Ki = 5128.61 nM T67162 CAQ6I5 137636351 Ki = 0.3 nM T67162 CFM92C 137636384 Ki = 6698 nM T67162 C6GWQ3 137636460 Ki = 36 nM T67162 CQ20FO 137636498 Ki = 1.5 nM T67162 CZU6N5 137636581 Ki = 4500 nM T67162 C0YDQ5 137637428 Ki = 1500 nM T67162 C8U7ZW 137637481 Ki = 121 nM T67162 CF7KG5 137637817 Ki = 6168 nM T67162 CDX39B 137637994 Ki = 1011 nM T67162 CXO70S 137638203 Ki = 60.6 nM T67162 CPQ98N 137638817 Ki = 1500 nM T67162 C49VDK 137638973 EC50 = 0.16 nM T67162 CA03VC 137639125 Ki = 104.71 nM T67162 C1HX3Z 137639304 Ki = 8900 nM T67162 C51HEL 137639330 Ki = 588 nM T67162 CC16HE 137640152 Ki = 350 nM T67162 CZP68A 137640189 Ki = 0.67 nM T67162 CZ4TA9 137640201 Ki = 912.01 nM T67162 CB2NO0 137640203 Ki = 7.4 nM T67162 CV49MZ 137640371 EC50 = 0.12 nM T67162 CN4ST6 137640376 Ki = 37579 nM T67162 CCU7L3 137640391 Ki = 0.55 nM T67162 C1EK3W 137640451 Ki = 9792 nM T67162 CX4A3N 137640511 Ki = 4466.84 nM T67162 C3U5NF 137640522 IC50 = 7.8 nM T67162 C8IO0R 137640836 Ki = 19 nM T67162 CWQ80N 137640967 IC50 = 9.44 nM T67162 CI1TU3 137641550 Ki = 124 nM T67162 CWXF83 137641643 Ki = 60152 nM T67162 C3LYX9 137641832 Ki > 10000 nM T67162 C4I6QS 137641944 IC50 = 2.87 nM T67162 C6PT7L 137642033 Ki = 35 nM T67162 C5WS6Q 137642134 Ki = 418 nM T67162 C94WSH 137642380 Ki = 7.8 nM T67162 C4Q6ZM 137642607 Ki = 457.09 nM T67162 CPX85V 137642676 Ki = 493 nM T67162 CUT21E 137642921 Ki = 73 nM T67162 CAC6W0 137643122 Ki = 1.1 nM T67162 C71XIQ 137643132 Ki = 200 nM T67162 CK51LB 137643309 EC50 = 0.11 nM T67162 CMJU75 137643395 IC50 = 11.8 nM T67162 C3O0FX 137643951 Ki = 1.4 nM T67162 CK5HG6 137644041 Ki = 17.7 nM T67162 C0HS3L 137644131 Ki = 9500 nM T67162 CWUM83 137644521 Ki > 10000 nM T67162 CDA80E 137644790 Ki = 145 nM T67162 C34PUI 137644833 Ki = 5.1 nM T67162 C0KL6Q 137644962 Ki = 3801.89 nM T67162 CVX6T1 137644966 Ki = 0.52 nM T67162 C4PV8U 137645196 Ki = 3400 nM T67162 CHT42S 137645295 IC50 = 80 nM T67162 CPCY48 137645406 IC50 = 1616 nM T67162 CZ8CU6 137645501 Ki = 149 nM T67162 CNH95X 137645574 Ki = 0.89 nM T67162 C3TP2G 137645830 Ki = 68 nM T67162 C2L4CG 137645834 Ki = 19.9 nM T67162 CCP38D 137645926 Ki = 141 nM T67162 CG8P6I 137645938 Ki = 524.81 nM T67162 CVX74E 137646045 Ki = 1489 nM T67162 C96EAP 137646245 Ki = 15.49 nM T67162 CPI68E 137646281 EC50 = 254 nM T67162 C8PV0N 137646568 IC50 = 7.6 nM T67162 C8C7UI 137647058 Ki = 34.7 nM T67162 C1C3YT 137647150 Ki = 202 nM T67162 CYH5U9 137647533 Ki = 37 nM T67162 CO5U9A 137647674 IC50 = 875 nM T67162 CWY02V 137648255 Ki = 317 nM T67162 C5XL4K 137648359 Ki = 940 nM T67162 C0X4WB 137649193 Ki = 114945 nM T67162 CVYC51 137649540 Ki = 21216 nM T67162 C75ELQ 137649585 Ki = 21.8 nM T67162 C3IF6W 137649770 EC50 = 104.5 nM T67162 CSPE25 137649896 Ki = 133 nM T67162 CMXI62 137649997 Ki = 1237 nM T67162 CB4HG5 137650482 IC50 = 36.6 nM T67162 CWQF69 137650550 IC50 = 10.4 nM T67162 C52IRM 137650705 Ki = 76 nM T67162 CFBL16 137650746 Ki = 8.41 nM T67162 C6R3IG 137650900 Ki = 57101 nM T67162 CKG08R 137650961 Ki = 1821 nM T67162 CR3Z6M 137651073 Ki = 12 nM T67162 CW4T6D 137651322 Ki = 0.73 nM T67162 C47TWK 137651544 IC50 = 37.6 nM T67162 CS3OV1 137651866 Ki = 6370 nM T67162 CU4S1W 137651887 Ki = 5.5 nM T67162 C15YDU 137651936 EC50 = 0.12 nM T67162 CVK26R 137652044 Ki = 1218 nM T67162 CC9F7J 137652174 EC50 = 135 nM T67162 CHFK13 137652210 Ki = 5162 nM T67162 C51CGJ 137652310 Ki = 223 nM T67162 CS61YC 137652312 Ki = 83671 nM T67162 C94NAQ 137652404 Ki = 190 nM T67162 CU8E4M 137652517 Ki = 23.8 nM T67162 C65RCN 137653034 Ki = 8.43 nM T67162 CX30HQ 137653096 Ki = 5700 nM T67162 C5ZJN8 137653359 Ki = 306 nM T67162 C32FLB 137653517 Ki = 10 nM T67162 C04XYN 137653567 IC50 = 3.29 nM T67162 CQ93DX 137653577 Ki = 1842 nM T67162 C2E3FV 137653850 Ki = 37 nM T67162 C48VDP 137653978 Ki = 54.8 nM T67162 C4C6EV 137653986 Ki = 1800 nM T67162 COTX19 137654511 Ki = 250 nM T67162 C6N0DT 137654586 IC50 = 5 nM T67162 CX82HS 137654666 Ki = 0.7 nM T67162 CF5Y2A 137654675 Ki = 3.7 nM T67162 C0SKV1 137654850 Ki > 10000 nM T67162 CLI4D8 137655029 Ki = 2.9 nM T67162 C4VG0U 137655411 Ki = 30 nM T67162 C7RW9H 137655451 EC50 = 1.5 nM T67162 CJAZ13 137655556 Ki = 46 nM T67162 C6CA5H 137655594 Ki = 480 nM T67162 CUC54G 137655636 Ki = 288.4 nM T67162 CDAN02 137655735 Ki = 0.52 nM T67162 CD16SQ 137655795 Ki = 2.2 nM T67162 CMA0T6 137655799 Ki = 29300 nM T67162 CXH16S 137655884 Ki = 273 nM T67162 CI68MV 137655953 EC50 = 3.1 nM T67162 CLT53E 137656298 Ki = 93.1 nM T67162 CVEN03 137656381 IC50 > 10000 nM T67162 CJO23S 137656836 Ki = 2290 nM T67162 CO3L7F 137656918 Ki > 10000 nM T67162 CA7F5N 137657115 Ki = 1.9 nM T67162 CV2CR4 137657153 EC50 = 1.7 nM T67162 C1HA0D 137657276 Ki = 316 nM T67162 CE0Y7P 137657322 Ki = 0.58 nM T67162 CRT86S 137657427 Ki = 0.81 nM T67162 CME6U8 137657882 EC50 = 0.0955 nM T67162 CEJ9L8 137657949 IC50 = 26.7 nM T67162 CH76FP 137657951 Ki = 200 nM T67162 CY4H6C 137658100 EC50 = 14.7 nM T67162 C3LHT5 137658253 IC50 = 40.5 nM T67162 C8G0HO 137658832 IC50 = 27 nM T67162 CFQ7C9 137659145 IC50 = 8.29 nM T67162 CEZ07P 137659303 Ki = 5.8 nM T67162 CT9YA5 137659335 Ki = 104847 nM T67162 CLQX32 137659728 IC50 = 9.65 nM T67162 CG2U9R 137659809 Ki = 140 nM T67162 CP9AN6 137659990 EC50 = 0.17 nM T67162 CP6US4 137660046 Ki = 0.86 nM T67162 CF9RZ5 137660385 IC50 = 20 nM T67162 C8W3AQ 137660395 Ki = 38.7 nM T67162 C5V4DQ 137660707 Ki = 2 nM T67162 CX4D7Y 137660741 Ki = 148 nM T67162 C1VB2N 137660751 Ki = 284 nM T67162 C42IDE 137660837 EC50 = 0.11 nM T67162 CG8QR9 137660855 Ki = 476 nM T67162 CDA8V2 137661377 Ki = 912.01 nM T67162 C5X9LH 137661635 EC50 = 53 nM T67162 CZI74G 137661939 Ki = 7501 nM T67162 CT3P2B 137662048 Ki > 109574 nM T67162 C9YXI5 137662136 Ki = 111 nM T67162 C0R6XM 138691314 Ki = 4847 nM T67162 CU3Y7W 138691316 Ki > 10000 nM T67162 CH2W4P 138691317 Ki > 10000 nM T67162 CHSC40 138691321 Ki = 3020 nM T67162 C18UZA 138691329 Ki > 10000 nM T67162 C1XWV0 138691338 Ki > 10000 nM T67162 C6LE1A 138691362 Ki > 10000 nM T67162 CN9R4A 138691364 Ki > 10000 nM T67162 C8H2KR 138691366 Ki > 10000 nM T67162 C2Z9CD 139488518 Ki > 10000 nM T67162 CJK95T 139488527 Ki > 10000 nM T67162 CZ6H9M 139488539 Ki > 10000 nM T67162 CAF2H8 139488606 Ki = 7080 nM T67162 C54CIL 139488740 Ki > 10000 nM T67162 CH7Y5D 141312275 Ki = 142 nM T67162 C7WJT2 142573371 Ki = 3250 nM T67162 CT3SY0 142573376 Ki = 26739 nM T67162 C9B0JX 142573379 Ki = 13904 nM T67162 CQO6K2 142573380 Ki = 9248 nM T67162 CEXL42 142573384 Ki = 6379 nM T67162 CJIC89 142573385 Ki = 1162 nM T67162 CAL25K 142573386 Ki = 12137 nM T67162 C5BOX1 142573395 Ki = 5165 nM T67162 CX6S8U 142573399 Ki = 12584 nM T67162 CIZ75U 142573404 Ki = 5650 nM T67162 CXI8C3 142573405 Ki = 3762 nM T67162 CG2H3O 142573406 Ki = 65229 nM T67162 C1L0GO 142573412 Ki = 2112 nM T67162 CCY49O 142573415 Ki = 48584 nM T67162 CFX0W5 142573417 Ki = 98462 nM T67162 C09XCG 142573420 Ki = 26253 nM T67162 C1IBV7 142573422 Ki = 1574 nM T67162 CQ0E4W 142573428 Ki = 2766 nM T67162 CB5M2G 142573431 Ki = 197 nM T67162 CNZX48 142573438 Ki = 21172 nM T67162 CQ5W7B 142573439 Ki = 25823 nM T67162 C7G3NO 142573444 Ki = 5891 nM T67162 CN5WK4 142573449 Ki = 9004 nM T67162 CORZ59 145948563 EC50 = 1380.38 nM T67162 CO5DR9 145949220 Ki = 782 nM T67162 CWAF96 145949371 Ki = 267 nM T67162 CHG2W6 145950605 Ki = 1285 nM T67162 COU57L 145950881 Ki = 506 nM T67162 CD4M6B 145951915 Ki = 269 nM T67162 C78AUI 145952711 Ki = 601 nM T67162 C0JO8B 145954831 Ki = 1033 nM T67162 CHI1V8 145956064 Ki = 497 nM T67162 CSER68 145956892 Ki = 366 nM T67162 CLVI07 145957637 Ki = 301 nM T67162 C91IDE 145958490 Ki = 534 nM T67162 C8VS7K 145959257 Ki = 931 nM T67162 CSIZ31 145959706 Ki = 1690 nM T67162 C85BSY 145963127 Ki = 5947 nM T67162 C4Y1PK 145963314 Ki = 1165 nM T67162 CEN94V 145963961 IC50 = 11.4 nM T67162 C3I6YP 145963975 IC50 = 123 nM T67162 C1B8QW 145964299 IC50 = 59.8 nM T67162 C95NZO 145964427 IC50 = 78.5 nM T67162 C0N8KC 145964622 IC50 = 53.5 nM T67162 C6T4RY 145964846 Ki = 299 nM T67162 C7MBS0 145964982 IC50 = 51.7 nM T67162 C7JS9I 145965041 IC50 = 412 nM T67162 C9D8IB 145965203 IC50 = 17.7 nM T67162 CV07EO 145965433 IC50 = 65.5 nM T67162 CJNG10 145966311 Ki = 250 nM T67162 CLM10C 145966333 IC50 = 24 nM T67162 C5L4WF 145967359 IC50 = 37.6 nM T67162 CL58XS 145967572 Ki = 368 nM T67162 C58WSL 145967904 Ki = 3555 nM T67162 CB1FD8 145968810 Ki = 343 nM T67162 CM6HG9 145968927 IC50 = 42.6 nM T67162 C2A0FO 145969167 IC50 = 59 nM T67162 C48XNG 145969667 Ki = 42 nM T67162 CNZY06 145969934 Ki = 369 nM T67162 C61MSO 145970938 Ki > 10000 nM T67162 CRC9T0 145971556 IC50 = 26.5 nM T67162 CR06QO 145972382 IC50 = 42.5 nM T67162 CWRM23 145972513 IC50 = 11.4 nM T67162 CEOY46 145973577 Ki = 1206 nM T67162 CL74IP 145973853 Ki = 303 nM T67162 CR0CX6 145974087 Ki = 876 nM T67162 C6AGN3 145974143 IC50 = 89.1 nM T67162 CW6EX3 145974189 Ki = 328 nM T67162 CDOJ39 145974939 IC50 = 8 nM T67162 CR83MU 145975214 IC50 = 51.1 nM T67162 CJF4Z0 145975393 IC50 = 9.3 nM T67162 CZ39GQ 145975595 IC50 = 299 nM T67162 C8XFM7 145976120 Ki = 4963 nM T67162 CCDU50 145976348 IC50 = 85 nM T67162 C34XME 145976696 IC50 = 82 nM T67162 C9FR7N 145976732 IC50 = 86.1 nM T67162 C72SMR 145978208 IC50 = 65.2 nM T67162 C1Q2BR 145978965 IC50 = 14.1 nM T67162 C20XQJ 145979626 Ki = 10080 nM T67162 C87MSW 145980271 Ki = 550 nM T67162 CW2CO4 145980458 Ki = 295 nM T67162 C8I7QL 145980875 Ki = 460 nM T67162 C4AF0G 145981310 IC50 = 28 nM T67162 C67AIW 145981408 IC50 = 5.3 nM T67162 C3N5DH 145981580 Ki = 860 nM T67162 COY79P 145982165 Ki = 256 nM T67162 CO7WP6 145982353 IC50 = 9.4 nM T67162 CEK60A 145982506 Ki = 42 nM T67162 CNE72W 145982756 EC50 = 7.6 nM T67162 CI59TX 145983018 Ki = 9 nM T67162 CYC58R 145983059 Ki = 24 nM T67162 CE2HG1 145983104 Ki = 45 nM T67162 C4F5OT 145983128 Ki = 8 nM T67162 C5ZG9M 145983139 Ki = 4 nM T67162 CV2GU9 145983144 Ki = 11 nM T67162 CWI9T1 145983268 Ki = 94 nM T67162 C4PKM2 145983390 Ki = 3 nM T67162 CIAF74 145983468 Ki = 11 nM T67162 CE7MF4 145983751 Ki = 5 nM T67162 CDQ4U7 145983760 Ki = 10 nM T67162 CO84BZ 145983763 Ki = 252 nM T67162 CYW9B2 145983794 Ki = 23 nM T67162 C1DW4U 145983928 IC50 = 6.4 nM T67162 C8I1WG 145983961 Ki = 0.9 nM T67162 CP5H4D 145984065 Ki = 12 nM T67162 C58DHN 145984151 IC50 = 213 nM T67162 CJ35DM 145984299 Ki = 0.14 nM T67162 C1RI8D 145984337 Ki = 251 nM T67162 CXTG03 145984446 Ki = 186 nM T67162 CXU69G 145984484 EC50 = 3.3 nM T67162 CU7E4M 145984511 Ki = 10 nM T67162 C6JUY0 145984737 Ki = 0.5 nM T67162 CID02G 145984807 Ki = 5 nM T67162 CM5X3V 145985050 Ki = 0.1 nM T67162 CG10LK 145985224 Ki = 4 nM T67162 CFJ9B3 145985233 Ki = 1.7 nM T67162 C5AOI6 145985289 Ki = 6 nM T67162 CC5KA9 145985295 EC50 = 5.5 nM T67162 CW30NA 145985505 Ki = 3 nM T67162 C7ZRP1 145985527 Ki = 15 nM T67162 C2XY8Q 145985533 Ki = 1 nM T67162 C7NI4X 145985585 Ki = 3 nM T67162 C9LJ5T 145985692 Ki = 0.3 nM T67162 C7QIX0 145985718 Ki = 7 nM T67162 C6V5QS 145985823 Ki = 2 nM T67162 C8F4JV 145985945 Ki = 115 nM T67162 C07GKD 145985958 Ki = 12 nM T67162 CCM18E 145986031 Ki = 21 nM T67162 CR0XQ3 145986138 Ki = 29 nM T67162 C2KGY7 145986176 EC50 = 3 nM T67162 CP6DT9 145986441 Ki > 10000 nM T67162 CXC79K 145986552 IC50 = 543 nM T67162 CT37DW 145986720 Ki = 1152 nM T67162 CNJH37 145986752 Ki = 417 nM T67162 C3VN5O 145987559 Ki = 4353 nM T67162 CZ5O8R 145987659 IC50 = 32.4 nM T67162 COS58J 145987942 IC50 = 2.5 nM T67162 C6MHU2 145988006 IC50 = 44.6 nM T67162 CHOB70 145988038 IC50 = 7.2 nM T67162 CO4LK7 145988180 Ki = 464 nM T67162 C9W1QA 145988497 IC50 = 13 nM T67162 CUGO10 145988693 Ki = 148 nM T67162 C9D2OG 145988738 Ki = 264 nM T67162 C4C0YP 145988913 Ki = 4116 nM T67162 CVC14L 145989181 IC50 = 80.2 nM T67162 CR2EV8 145989183 IC50 = 80.6 nM T67162 CMJL94 145989451 IC50 = 2 nM T67162 CBN7D9 145990000 Ki = 202.3 nM T67162 C3GPR9 145990093 Ki = 20030 nM T67162 C41SBL 145990126 IC50 = 4.3 nM T67162 CLF26V 145990141 Ki = 1100 nM T67162 C6NYE9 145990254 Ki > 23889 nM T67162 C2Q5UK 145990353 Ki = 153 nM T67162 CPW28Y 145990453 Ki = 700 nM T67162 CT7AB8 145990459 Ki = 5233 nM T67162 CE9PT1 145990482 IC50 = 9.6 nM T67162 CMJ46R 145990794 IC50 = 6.1 nM T67162 C5TNP0 145991127 IC50 = 38.1 nM T67162 CW14AE 145991244 IC50 = 8.4 nM T67162 CU6E1Z 145991746 IC50 = 119 nM T67162 CB8CM6 145992305 Ki = 3429 nM T67162 CCP2U1 145992489 Ki = 317 nM T67162 CELG57 145992523 IC50 = 30.1 nM T67162 CLPU06 145992567 Ki = 273 nM T67162 CB64KH 145992860 IC50 = 9.8 nM T67162 C9PS8N 145993117 IC50 = 10.9 nM T67162 CT63XO 145993172 IC50 = 8.5 nM T67162 CRWE54 145993377 Ki = 800 nM T67162 C0Z6YX 145993493 IC50 = 24.4 nM T67162 C17HSV 145993577 IC50 = 11 nM T67162 C0TL8E 145993714 Ki = 416 nM T67162 C4TY6L 145993896 Ki = 2163.1 nM T67162 CC2G1V 146025727 Ki = 8700 nM T67162 CI9GM7 146025765 EC50 = 6.761 nM T67162 CQ21OZ 146025766 EC50 = 46.77 nM T67162 CV3U7W 146025767 EC50 = 70.79 nM T67162 CH3VY4 146025768 EC50 = 14 nM T67162 CLD9A6 146025769 EC50 = 7.586 nM T67162 CR4Q5F 146025770 EC50 = 131.83 nM T67162 CXQ2H1 146025774 EC50 = 2 nM T67162 C6S9PX 146025775 EC50 = 9.772 nM T67162 CC8E2M 146025776 EC50 = 2.818 nM T67162 C4F9AT 146025777 EC50 = 5 nM T67162 CS05BD 146025778 EC50 = 4.786 nM T67162 C9G4IM 146025779 EC50 = 0.4 nM T67162 CPQ26G 146025780 EC50 = 67 nM T67162 C1EAO0 146025781 EC50 = 128.82 nM T67162 CHBX23 146025782 EC50 = 26.92 nM T67162 CF7E6W 146025783 EC50 = 85.11 nM T67162 CZI83F 146025784 EC50 = 19 nM T67162 CEY6N7 146025811 IC50 = 0.123 nM T67162 CZO92Q 146025812 IC50 = 337.5 nM T67162 CY97RS 146025813 IC50 = 44.67 nM T67162 C6NGR9 146025814 IC50 = 1949.84 nM T67162 CXNT51 146025815 IC50 = 28.18 nM T67162 C7O0GT 146025816 IC50 = 40.74 nM T67162 CC1UL6 146025817 EC50 = 2561 nM T67162 C6IOM8 146025818 EC50 = 1258.93 nM T67162 CT3I4V 146025819 EC50 = 602.56 nM T67162 CJ9I7W 146025820 EC50 = 575.44 nM T67162 CSL0Q5 146025821 EC50 = 1621.81 nM T67162 CRJ3Z7 146025822 EC50 > 10000 nM T67162 C9FY3J 146025823 EC50 > 10000 nM T67162 CO9A5N 146451658 Ki = 424 nM T67162 C12RYJ 146451661 Ki = 1440 nM T67162 C9MCB1 146451664 Ki = 537 nM T67162 C65FZJ 146451691 Ki = 364 nM T67162 C5ZOJ3 146680920 Ki = 3319 nM T67162 COQF36 149438247 IC50 = 1200 nM T67162 CU9FD3 151880864 Ki = 26050 nM T67162 C6P3SR 153287553 Ki > 10000 nM T67162 CV9G7Z 153287572 Ki > 10000 nM T67162 CO85KL 153287574 Ki > 10000 nM T67162 CQKH93 154395193 Ki = 1 nM T67162 CA9S3Y 155195287 Ki = 9160 nM T67162 C7XIR5 155195305 Ki = 7730 nM T67162 CQ5WA9 155195311 Ki = 87.8 nM T67162 CCFR96 155195429 Ki = 245 nM T67162 C3S2EX 155195430 Ki = 3860 nM T67162 C0RQT6 155195433 Ki = 10100 nM T67162 CL61UG 155195435 Ki = 27000 nM T67162 C10GRK 155195439 Ki = 341 nM T67162 CME84G 155195441 Ki = 2510 nM T67162 CQ3G0P 155195442 Ki = 21100 nM T67162 CH4BL7 155195444 Ki = 5220 nM T67162 C1JQ7Y 155195448 Ki = 9450 nM T67162 CM9RP4 155195449 Ki = 120 nM T67162 CON51V 155195451 Ki = 6710 nM T67162 CL9Z5V 155195452 Ki = 34.6 nM T67162 CLQ72J 155195454 Ki = 5510 nM T67162 CUH20V 155195486 Ki = 831 nM T67162 CG5NW0 155195487 Ki = 106 nM T67162 CJK6C0 155195495 Ki = 8240 nM T67162 C6ZV8B 155195496 Ki = 134 nM T67162 CF3EY0 155195497 Ki = 6260 nM T67162 COJL79 155195501 Ki = 113 nM T67162 CD2EV4 155195516 Ki = 2660 nM T67162 CZ1K4D 155510674 Ki = 15 nM T67162 C3MC0Q 155510756 Ki = 19 nM T67162 CC3KP7 155510927 Ki = 1202 nM T67162 C5DQG2 155510939 IC50 > 10000 nM T67162 CM4RB0 155511262 Ki = 391 nM T67162 C13IEH 155511416 Ki = 2754.23 nM T67162 CTW28Q 155511803 Ki > 50000 nM T67162 CA0LF6 155511820 Ki = 0.4467 nM T67162 C9KX6O 155511928 Ki = 336 nM T67162 CJ96WB 155512259 Ki = 46 nM T67162 C1YB7P 155512384 Ki = 41686.94 nM T67162 CXF90M 155512487 Ki = 376 nM T67162 CQ83KZ 155512662 Ki = 743 nM T67162 C2TRB6 155512841 Ki = 14.7 nM T67162 C0DKF9 155512851 Ki = 757 nM T67162 CO68LC 155512944 Ki > 10000 nM T67162 C6XST7 155513053 Ki = 1159 nM T67162 C6FEW4 155513265 Ki > 20000 nM T67162 C35GHL 155513375 Ki = 16318 nM T67162 CD4Y8Z 155513529 Ki = 2511.89 nM T67162 C36RDV 155513614 Ki = 950 nM T67162 C0ZXT4 155513773 Ki = 34 nM T67162 CHXY56 155513802 Ki = 4823 nM T67162 CL5G9Q 155513837 Ki = 537 nM T67162 CX7A3L 155513965 Ki = 18.2 nM T67162 CF6K8R 155514137 Ki = 620 nM T67162 C7FI9W 155514217 Ki = 28 nM T67162 C95QOT 155514378 Ki = 302 nM T67162 CK9YN0 155514430 Ki = 29.8 nM T67162 C3SQI7 155514459 Ki > 10000 nM T67162 CI4DT8 155514575 Ki = 87 nM T67162 CJUI87 155514774 Ki = 9 nM T67162 CH34RK 155514798 Ki > 5000 nM T67162 C5AM4N 155514868 Ki = 29.51 nM T67162 CV8F7A 155515301 Ki = 2187.76 nM T67162 C3NB0D 155515324 Ki = 50140 nM T67162 C0Q8PR 155515407 Ki = 204 nM T67162 CWO56B 155515415 Ki > 10000 nM T67162 C3XZM2 155515759 Ki = 110 nM T67162 C2TN5D 155515890 Ki = 867 nM T67162 CUE5J3 155515907 Ki = 3144 nM T67162 C7KT0D 155515919 Ki = 1318 nM T67162 CM65NQ 155515931 Ki = 47 nM T67162 C13LOV 155515942 Ki = 1410 nM T67162 CAS50P 155515966 Ki = 27359 nM T67162 CUM2N4 155515982 Ki = 73 nM T67162 CV12SD 155516041 Ki = 550 nM T67162 C7OF4C 155516118 Ki = 505 nM T67162 CJ98ZK 155516236 Ki = 1161.4 nM T67162 CG5M1O 155516282 Ki = 180 nM T67162 CH7N0C 155516494 Ki = 46260 nM T67162 CQY58Z 155516873 Ki = 440 nM T67162 CEA9D5 155517238 Ki = 141 nM T67162 C9ZAW0 155517266 Ki > 5000 nM T67162 C47LRQ 155518026 Ki = 110 nM T67162 CW0B5K 155518159 Ki > 10000 nM T67162 C79MXU 155518617 Ki = 12046 nM T67162 CYB12O 155518974 Ki = 40040 nM T67162 CCEZ93 155519102 Ki = 1001 nM T67162 CPER92 155519378 Ki = 94 nM T67162 CQD2J7 155519393 Ki = 1025 nM T67162 C2SXT1 155519515 Ki = 304 nM T67162 C0KLD8 155519559 Ki = 240 nM T67162 C07BTO 155519598 Ki = 496 nM T67162 CUSA24 155519891 Ki > 10000 nM T67162 C8IYD1 155520455 Ki = 844.6 nM T67162 C5FL7R 155520499 Ki = 264 nM T67162 C8OC3W 155520552 Ki = 220 nM T67162 C5DSE0 155520996 Ki = 380.2 nM T67162 C17QKW 155521049 Ki = 148 nM T67162 CQ76MP 155521503 Ki = 2344 nM T67162 C7SG3T 155521675 Ki = 151.36 nM T67162 C9R5AM 155521711 Ki = 169 nM T67162 C1OS6D 155522116 Ki = 3981 nM T67162 C98RDQ 155522218 Ki = 17670 nM T67162 C5NM0F 155522454 EC50 = 2.09 nM T67162 C2TV4Y 155522487 Ki > 10000 nM T67162 CP6H1D 155522562 Ki = 121 nM T67162 CV7IG5 155522663 Ki = 512.9 nM T67162 CD59RE 155522719 Ki > 50000 nM T67162 C8B2WR 155522744 IC50 = 8810 nM T67162 CUG8L3 155522920 Ki > 10000 nM T67162 C2H3JL 155523073 Ki = 407.4 nM T67162 CQA76T 155523112 Ki = 3494 nM T67162 CUG4Q8 155523121 Ki = 3981 nM T67162 C3E9DJ 155523127 Ki > 5000 nM T67162 C50RNQ 155523337 Ki = 1.479 nM T67162 CG6Y4Z 155523515 Ki = 42 nM T67162 CD9QU6 155523519 Ki = 8 nM T67162 C2Y9CW 155523745 Ki = 151 nM T67162 CVQ68Y 155523770 Ki = 1083.9 nM T67162 COH1Q5 155524191 Ki = 676 nM T67162 C5KYB4 155524228 Ki = 20 nM T67162 CW7NT8 155524423 Ki = 1502 nM T67162 CK4B0R 155524491 Ki = 896 nM T67162 CUO93F 155524808 Ki = 113 nM T67162 CQB0M8 155524884 Ki = 3162 nM T67162 C65UZD 155524956 Ki = 142 nM T67162 CQX27T 155525357 Ki = 2105 nM T67162 CT0NV4 155525431 Ki > 50000 nM T67162 CT1YQ0 155525527 EC50 = 22.9 nM T67162 CR3DZ7 155525571 Ki = 321 nM T67162 CW65KS 155525705 Ki = 1116 nM T67162 CZ81JA 155526026 Ki = 45 nM T67162 CPZ0H7 155526424 Ki = 3449 nM T67162 C1U2XO 155526651 Ki = 82 nM T67162 C9ANR8 155527358 Ki = 19634 nM T67162 C9IW8F 155527714 Ki = 19 nM T67162 C3PS9Z 155527787 Ki = 299 nM T67162 CEQ8O4 155527891 Ki = 112 nM T67162 CGA2J9 155528048 Ki = 5495.41 nM T67162 CW68KC 155528355 Ki > 10000 nM T67162 C7C1EF 155528967 Ki = 963 nM T67162 C5J7AU 155529153 Ki = 656 nM T67162 CU69ZH 155529400 Ki = 2.818 nM T67162 C9KS5C 155529450 Ki = 7 nM T67162 CEN90X 155529453 Ki = 58 nM T67162 C1OAX6 155529543 Ki = 7.762 nM T67162 CUSG17 155529568 Ki = 140 nM T67162 C8U7QC 155529592 Ki = 30 nM T67162 CKZ25Y 155529679 Ki = 27 nM T67162 CBS2O8 155529683 Ki > 5000 nM T67162 C7UZI1 155530285 Ki = 3802 nM T67162 C3X4IA 155530328 Ki = 39 nM T67162 C9PC3D 155530350 Ki = 927 nM T67162 C8WC5Y 155530733 Ki = 71 nM T67162 CDGX72 155530763 EC50 = 50.1 nM T67162 CGC9N0 155530882 Ki = 2.4 nM T67162 C98YQF 155531012 Ki = 105 nM T67162 C4W6VC 155531065 Ki = 757 nM T67162 C71WHE 155531162 Ki = 169.82 nM T67162 C5HWP4 155531362 Ki > 10000 nM T67162 CQ86CH 155531455 Ki > 10000 nM T67162 C95JRV 155531663 EC50 = 9.3 nM T67162 C9YMR2 155531801 Ki = 132 nM T67162 C4VK0L 155531809 Ki = 490 nM T67162 CCT8V9 155531846 Ki = 1348 nM T67162 C3R4YM 155532148 Ki = 112.2 nM T67162 CKZ35G 155532475 Ki > 5000 nM T67162 C4LOR5 155532477 Ki > 5000 nM T67162 CK9JP0 155532505 Ki = 22 nM T67162 CX35QS 155532545 Ki > 10000 nM T67162 CKXC68 155532666 Ki = 0.84 nM T67162 C3W6HV 155532983 Ki = 5129 nM T67162 CX6DV4 155533028 Ki = 431 nM T67162 C23GDV 155533534 Ki = 1977 nM T67162 CSY06A 155533573 Ki = 5248 nM T67162 C3OEH2 155533648 Ki = 141 nM T67162 C15RYP 155533660 Ki > 10000 nM T67162 CZA89B 155533824 Ki = 58.1 nM T67162 CY01GZ 155533850 Ki = 1651 nM T67162 CQ12KS 155533996 Ki = 4606 nM T67162 CP3J8B 155534152 Ki = 1585 nM T67162 C3L0CP 155534184 Ki > 10000 nM T67162 C8AX5N 155534186 Ki > 5000 nM T67162 CA2LG1 155534225 Ki = 19.05 nM T67162 CZTX89 155534246 Ki = 23 nM T67162 CG85SB 155534301 Ki = 188 nM T67162 C3VGT0 155534362 Ki = 1129 nM T67162 CW7SV9 155534575 Ki = 51 nM T67162 C75FSY 155534794 Ki = 1175 nM T67162 CC4D5K 155535057 Ki = 0.844 nM T67162 C6KF4E 155535154 Ki = 1802 nM T67162 C71YMQ 155535169 Ki = 138 nM T67162 CGZ5T8 155535272 Ki = 2.93 nM T67162 C3V1CL 155535404 Ki > 225748 nM T67162 CA3N2X 155535680 Ki = 6309.57 nM T67162 CEZ46A 155535732 Ki = 2.455 nM T67162 C4LDC6 155535761 Ki = 1.514 nM T67162 CHP2Z9 155535866 Ki = 3162 nM T67162 C14JEX 155535878 Ki = 708 nM T67162 CA01QX 155536022 Ki = 210 nM T67162 C0QA4L 155536040 Ki = 3.548 nM T67162 CB79ZW 155536080 Ki > 10000 nM T67162 C5I1JA 155536087 Ki = 24 nM T67162 C72FLG 155536152 Ki = 1234 nM T67162 CDL9R5 155536374 Ki = 186 nM T67162 CYB1F2 155536713 Ki = 11.22 nM T67162 CDEX60 155536720 Ki = 200 nM T67162 CY61EO 155536815 Ki = 7824 nM T67162 C7FVE8 155537034 Ki = 5561 nM T67162 C36FRH 155537074 Ki = 178 nM T67162 CD75GP 155537227 Ki > 10000 nM T67162 CFCG03 155537361 Ki = 24 nM T67162 C6NT4F 155537490 Ki = 177.83 nM T67162 CVFD68 155537516 Ki = 1349 nM T67162 CBF8K6 155537861 Ki = 3.548 nM T67162 C13CSU 155537907 Ki = 216 nM T67162 CP3WK6 155538028 Ki = 180 nM T67162 CB8IC7 155538144 Ki > 10000 nM T67162 C2S9LF 155538235 Ki = 21098 nM T67162 C5F2GI 155538236 Ki = 2349 nM T67162 CFPT03 155538349 Ki = 520 nM T67162 C9TIU2 155538367 Ki = 9333 nM T67162 C75SRB 155538429 Ki = 261 nM T67162 C83KQL 155538443 IC50 = 500 nM T67162 CYC1P3 155538451 Ki = 27 nM T67162 CM08NT 155538716 Ki > 10000 nM T67162 CQ69UA 155538814 Ki = 674 nM T67162 C3DIY2 155539246 Ki = 253.1 nM T67162 CAOV97 155539413 Ki = 35720 nM T67162 CAT98F 155539483 Ki = 19 nM T67162 CPV48W 155539557 Ki = 323.6 nM T67162 C6S8BA 155539600 Ki = 520 nM T67162 C7T1EF 155539653 IC50 = 15 nM T67162 C42GUK 155540147 Ki > 10000 nM T67162 CJD9C8 155540541 Ki = 411 nM T67162 C19GLX 155540715 Ki = 112.2 nM T67162 C2OWD4 155540721 Ki = 3631 nM T67162 CR2K1T 155540795 Ki = 1622 nM T67162 CNU92V 155540807 Ki = 16 nM T67162 C8WRH2 155540919 Ki = 56 nM T67162 COS2E7 155541072 Ki > 10000 nM T67162 CMP8Q2 155541547 Ki = 2138 nM T67162 C0D5ZP 155541775 EC50 = 330 nM T67162 C9CQI3 155541844 Ki = 21.88 nM T67162 CP7UG2 155541866 Ki = 1365 nM T67162 COZ46W 155541871 Ki = 75 nM T67162 C58YSH 155542160 Ki = 1592 nM T67162 CM9FI1 155542182 Ki = 120 nM T67162 C7U3JN 155542198 Ki = 245 nM T67162 CB62ZS 155542237 Ki = 1175 nM T67162 CXCW81 155542321 Ki = 1094 nM T67162 C9FS3Y 155542461 Ki > 10000 nM T67162 C18OPI 155542619 Ki = 257 nM T67162 CC51DL 155542687 Ki > 30000 nM T67162 CVK2M9 155543189 Ki = 4012 nM T67162 CDO05U 155543223 Ki = 355 nM T67162 CT6HY4 155543250 Ki = 1862 nM T67162 C3UXC2 155543605 IC50 > 100000 nM T67162 C68MSK 155543653 Ki = 566 nM T67162 C4ANI0 155543691 Ki = 1023 nM T67162 CIEQ43 155543869 Ki = 84 nM T67162 CZ7O0A 155544139 Ki = 1224 nM T67162 C08FTE 155544239 Ki = 2362 nM T67162 CY57ZS 155544392 Ki = 166 nM T67162 CD84VK 155544810 Ki = 58 nM T67162 CP62SB 155544891 Ki = 0.1585 nM T67162 C2XZD8 155545087 Ki = 254 nM T67162 CVB8S1 155545179 Ki = 1.023 nM T67162 CO9X1Z 155545526 Ki > 10000 nM T67162 CI0YL8 155545625 Ki > 10000 nM T67162 C74GFO 155546189 Ki = 90 nM T67162 CH3W9N 155546350 Ki > 10000 nM T67162 C7MCZ0 155546478 Ki = 507 nM T67162 C9D0GL 155547128 Ki = 51 nM T67162 C1SVX6 155547259 Ki = 211 nM T67162 CD02EN 155547436 Ki = 271 nM T67162 COJ27N 155547693 Ki = 740 nM T67162 CA9K1Y 155547729 Ki = 19655 nM T67162 CUGC98 155547873 Ki = 63.1 nM T67162 CECV12 155548038 Ki = 15768 nM T67162 CM4XB6 155548127 Ki = 180 nM T67162 CJ7AL8 155548205 Ki = 324 nM T67162 C9GM0D 155548336 Ki = 390 nM T67162 CHJ1C7 155548481 Ki = 29.51 nM T67162 C5LYE8 155548677 Ki = 167 nM T67162 C87JGN 155549153 Ki > 10000 nM T67162 CGP8O5 155549315 Ki = 2 nM T67162 C3KXY1 155549528 Ki = 165 nM T67162 C52FRY 155549978 Ki = 48 nM T67162 C0DHX7 155550192 Ki = 29 nM T67162 CN6I4P 155550431 Ki = 5934 nM T67162 C3Y1EJ 155550445 Ki = 4753 nM T67162 CY34NR 155550580 Ki = 310 nM T67162 C6N9PG 155550640 Ki = 5623 nM T67162 CG7NR9 155550756 Ki > 5000 nM T67162 C8HPN7 155551113 Ki = 320 nM T67162 C82QWR 155551173 Ki = 408 nM T67162 CY2P8T 155551269 Ki = 2.2 nM T67162 C61IVC 155551353 Ki > 10000 nM T67162 CHS71N 155551685 Ki = 132 nM T67162 C5RZ4U 155552000 IC50 = 280 nM T67162 C6E9LK 155552054 Ki = 114 nM T67162 CX8JA1 155552185 Ki = 110 nM T67162 CA1WS9 155552212 Ki = 94 nM T67162 C9T3AX 155552483 IC50 = 1080 nM T67162 CG70XQ 155552591 Ki > 5000 nM T67162 C63VOX 155552609 Ki = 1.1 nM T67162 CB4F8Y 155552676 Ki = 1502 nM T67162 C0DQ3Z 155552695 Ki = 233 nM T67162 CDQ7C2 155552798 Ki = 945 nM T67162 CPV35U 155552826 Ki > 10000 nM T67162 CP6KN4 155553364 Ki = 24994 nM T67162 C1RLI0 155553370 Ki > 10000 nM T67162 CN3Z2Q 155553911 Ki >= 17000 nM T67162 C3A2QG 155554001 Ki = 63.1 nM T67162 CD5LC6 155554006 Ki = 1421 nM T67162 CDV6B9 155554036 Ki = 2362 nM T67162 CKF75H 155554324 Ki = 197 nM T67162 CINW85 155554326 Ki = 61 nM T67162 C6ZSU3 155554462 Ki = 734 nM T67162 CRY82F 155554955 Ki = 1826 nM T67162 CELU08 155555060 Ki = 62 nM T67162 CWY29E 155555201 Ki = 1.86 nM T67162 C1RCM0 155555224 Ki = 136 nM T67162 C17XSQ 155555298 IC50 = 4940 nM T67162 C2E5TR 155555506 Ki = 368 nM T67162 C76IMR 155555589 Ki = 66 nM T67162 CYP63A 155556311 Ki = 26.9 nM T67162 CO52HW 155556527 Ki > 10000 nM T67162 C1I5JR 155556665 Ki = 59994 nM T67162 C5QYS0 155557134 Ki = 30 nM T67162 CXN47Z 155557425 Ki = 465 nM T67162 CD2L3K 155557443 Ki > 10000 nM T67162 CER48T 155557500 Ki > 10000 nM T67162 CQ6YT5 155557645 Ki = 2630 nM T67162 C3UCM2 155557792 Ki = 323.59 nM T67162 CF6H3V 155558408 Ki = 4369 nM T67162 C36SYJ 155558844 Ki = 380 nM T67162 CGBZ63 155559617 Ki = 4.3 nM T67162 C06BZW 155559811 Ki = 438 nM T67162 C1U4ZL 155560181 Ki = 213.8 nM T67162 C60GZE 155560295 Ki = 310 nM T67162 CNF8Y0 155560484 Ki = 5.248 nM T67162 CD61BM 155560516 Ki = 38.6 nM T67162 CJ9R1T 155561102 Ki = 1042 nM T67162 C7OZM6 155561446 Ki = 1148 nM T67162 C2HF6P 155561581 Ki = 506 nM T67162 CD2L9R 155561779 Ki = 94 nM T67162 CG3RL0 155561845 IC50 = 190 nM T67162 CALB48 155561861 Ki = 2049 nM T67162 C5O8AU 155561865 Ki > 10000 nM T67162 CTZE48 155561895 Ki = 85.11 nM T67162 COL7N8 155561901 Ki > 10000 nM T67162 CL45NV 155561914 Ki = 161 nM T67162 CW7M1D 155561995 Ki = 1047 nM T67162 C93KWN 155562202 Ki = 10 nM T67162 CF89GP 155562328 Ki = 35 nM T67162 C2Z0HB 155562353 Ki = 2435.9 nM T67162 CRMC43 155562395 Ki > 10000 nM T67162 CO3C6L 155562423 Ki > 10000 nM T67162 C2EBQ1 155562463 Ki = 64.57 nM T67162 CO0Q7N 155562484 Ki = 0.1202 nM T67162 C5AI0S 155562519 Ki = 62 nM T67162 C5BQ8U 155562652 Ki = 11160 nM T67162 CH0PW5 155562681 Ki = 1832 nM T67162 CF6B4W 155562834 Ki = 118 nM T67162 CZ6IA2 155562918 Ki = 4247 nM T67162 CV4PM8 155562984 Ki = 92.9 nM T67162 CRCW25 155562997 Ki = 190 nM T67162 CBH14K 155563164 Ki > 10000 nM T67162 CG1L8E 155563286 Ki > 10000 nM T67162 C4IH5Z 155563301 Ki > 10000 nM T67162 C1KU5D 155563347 Ki = 22.39 nM T67162 C38WXS 155563374 Ki = 1168 nM T67162 C5KCZ1 155563589 EC50 = 37.7 nM T67162 C0INS4 155563826 Ki = 1230 nM T67162 CAZL19 155563950 Ki = 670 nM T67162 CU7JG9 155564308 Ki = 26 nM T67162 C54WIE 155564667 Ki = 4.65 nM T67162 C0UN4V 155564747 Ki = 238 nM T67162 C3OK2L 155565059 Ki = 108 nM T67162 CIB3R0 155565292 Ki = 42 nM T67162 C4OZ2X 155565438 Ki = 140 nM T67162 C51ORX 155565531 Ki = 4.2 nM T67162 CMH8I1 155565768 Ki > 5000 nM T67162 C2MIU5 155565813 Ki = 446 nM T67162 CYIG07 155566058 Ki = 110 nM T67162 C7P5VG 155566191 Ki = 220 nM T67162 C42DAE 155566238 Ki = 281.84 nM T67162 C0Y9RV 155566355 Ki = 190 nM T67162 CRJG23 155566403 Ki = 410 nM T67162 C7O6YP 155566439 Ki = 2916 nM T67162 CK20WA 155566662 Ki = 233 nM T67162 CU46EB 155566665 Ki > 10000 nM T67162 CEV3B9 155566852 Ki = 458 nM T67162 C67LAG 155566854 Ki = 794 nM T67162 CW1TN7 155566925 Ki > 10000 nM T67162 C6DPR8 155566974 Ki = 992 nM T67162 C46ZDJ 155567045 Ki = 8434 nM T67162 C6HS0F 155567118 IC50 = 6360 nM T67162 C41UWT 155567307 Ki = 11 nM T67162 CC5ZK3 155567742 Ki = 46.77 nM T67162 C4NX7P 155567775 Ki = 99.7 nM T67162 C95RAP 155567835 Ki = 660.7 nM T67162 C5A6YM 155567869 Ki = 2105 nM T67162 C8NO4X 155567971 Ki = 380 nM T67162 CA68TK 155568224 Ki = 329 nM T67162 C4EX7C 155568246 Ki = 217 nM T67162 CRX8J2 155568278 Ki = 286 nM T67162 CP03VZ 155568299 Ki = 7079 nM T67162 CQ5N6X 155568411 Ki > 50000 nM T67162 C7FR1Q 155568415 Ki = 74272 nM T67162 CHO2G1 155568612 Ki = 17595 nM T67162 CVU42Z 155568628 Ki = 95 nM T67162 CV24CW 155568676 Ki = 3494 nM T67162 C73ERT 155568786 Ki = 275.4 nM T67162 CXP3E4 155568794 Ki = 1730 nM T67162 CKG5M1 155568867 EC50 = 1965 nM T67162 CB5IP9 155569021 Ki = 246 nM T67162 C42JKO 155569198 Ki = 1230 nM T67162 C0CZK6 155569337 Ki > 10000 nM T67162 CP9V7M 155569396 Ki = 8710 nM T67162 C3ZNX6 155569414 Ki = 239 nM T67162 CZ8RV4 155569568 Ki = 571 nM T67162 C3N9VU 10251906 Ki > 500 nM T67162 CP9TR0 10324985 Ki = 22.01 nM T67162 CP2EI0 118725998 EC50 = 204 nM T67162 CC2GF1 118726019 EC50 > 100000 nM T67162 CFS9W4 118726022 EC50 > 100000 nM T67162 C9J5HY 16105548 Ki = 16 nM T67162 C4ZD3A 16105549 Ki = 12 nM T67162 CFMK68 3246545 Ki = 1.2 nM T67162 D00CDM 115107 Ki > 10000 nM T67162 D00CPI 22397846 Ki = 69 nM T67162 D00GSD 25107716 Ki = 142 nM T67162 D00HUV 9881815 Ki = 85.6 nM T67162 D00NQV 5041 Ki > 1000 nM T67162 D00SDJ 11237664 Ki = 246 nM T67162 D00YEB 25141414 Ki = 55.5 nM T67162 D01CGM 3033677 Ki = 62 nM T67162 D01CXD 10398175 Ki > 10000 nM T67162 D01ENR 2993172 Ki > 10000 nM T67162 D01JXM 46222048 Ki > 1000 nM T67162 D01KIH 44323762 Ki = 257.5 nM T67162 D01PYU 9821248 Ki = 500 nM T67162 D02BXA 238317 Ki > 10000 nM T67162 D02MVR 2761023 Ki = 200 nM T67162 D02NNS 9845181 Ki = 580 nM T67162 D02YDU 10420539 Ki > 20000 nM T67162 D02YSX 197033 Ki = 630.96 nM T67162 D03DET 10287730 Ki = 3162.28 nM T67162 D03GES 9995378 Ki = 3200 nM T67162 D03JOS 233952 Ki = 120 nM T67162 D03JOX 11311147 IC50 > 10000 nM T67162 D03KUH 57267 Ki = 0.086 nM T67162 D03NRJ 10871642 Ki > 1500 nM T67162 D03PAH 410747 Ki = 19.95 nM T67162 D03PYX 1219 Ki = 2.27 nM T67162 D03TDN 1342 IC50 > 1000 nM T67162 D03TPY 9885123 IC50 > 10000 nM T67162 D03VPS 16094676 Ki > 10000 nM T67162 D04AAI 45380179 Ki = 431 nM T67162 D04AZE 3277600 Ki < 31622.78 nM T67162 D04CPW 25139331 Ki = 21000 nM T67162 D04CTN 11074524 Ki = 68 nM T67162 D04JUJ 54456 Ki = 5400 nM T67162 D04MVL 3082625 Ki = 1070 nM T67162 D04PBA 10015867 Ki = 4.6 nM T67162 D04RBU 45486362 Ki = 47.5 nM T67162 D04TQF 11973927 Ki = 5000 nM T67162 D04TWX 9794475 EC50 > 10000 nM T67162 D05AIN 22397839 Ki = 35 nM T67162 D05BCJ 2779264 Ki = 8500 nM T67162 D05EQG 5265 IC50 = 0.0000000003 nM T67162 D05HMW 10705550 Ki = 15000 nM T67162 D05KUM 135446209 Ki = 9 nM T67162 D05NQX 9961911 Ki = 517 nM T67162 D05NZI 44348012 Ki = 0.2512 nM T67162 D05QJK 9816808 Ki = 79.8 nM T67162 D05UUW 210956 Ki = 21 nM T67162 D05XGR 6918647 Ki = 3981.07 nM T67162 D05XNR 10034684 IC50 = 1030 nM T67162 D05ZUX 44207909 Ki = 831.76 nM T67162 D06AIQ 107995 Ki = 4.2 nM T67162 D06BWZ 68678 Ki = 5.4 nM T67162 D06FUV 5311189 Ki = 8.5 nM T67162 D06HTJ 24866612 EC50 = 19.9 nM T67162 D06LQH 167715 IC50 = 0.000000001 nM T67162 D06NTB 30438 Ki = 5500 nM T67162 D06QGD 11357862 IC50 > 10000 nM T67162 D06VDN 443391 IC50 > 1000 nM T67162 D06WLB 9838216 Ki = 81.8 nM T67162 D07CZJ 44447998 Ki > 10000 nM T67162 D07ETF 9838960 Ki = 28 nM T67162 D07GBV 10091189 Ki = 350 nM T67162 D07GQP 11477180 Ki = 74 nM T67162 D07LRJ 5312149 Ki = 460 nM T67162 D07RPV 65490 IC50 = 7 nM T67162 D07RYR 44396235 Ki > 10000 nM T67162 D07UUQ 15508240 Ki = 6300 nM T67162 D07VBS 10425450 Ki = 251 nM T67162 D07ZOP 11470616 IC50 > 10000 nM T67162 D08CKM 9863250 Ki = 1584.89 nM T67162 D08CZT 9882067 Ki > 1600 nM T67162 D08JCU 44439386 Ki > 2000 nM T67162 D08TCX 11437461 Ki > 10000 nM T67162 D08UQU 24766199 Ki = 235 nM T67162 D09CFW 57377246 Ki = 100 nM T67162 D09CVG 449126 Ki > 1800 nM T67162 D09FTZ 10564794 Ki = 15000 nM T67162 D09HFT 44439376 Ki > 1000 nM T67162 D09MGF 11973811 Ki = 5000 nM T67162 D09PIN 3378093 Ki > 1000 nM T67162 D09PJF 44588498 Ki = 40.6 nM T67162 D09RPR 16737207 Ki > 10000 nM T67162 D09WBJ 10336538 Ki = 1310 nM T67162 D0A2BE 2780 Ki = 12 nM T67162 D0A7AK 11973810 Ki = 5000 nM T67162 D0AX0K 5615 IC50 = 620 nM T67162 D0B0UZ 9861462 Ki > 10000 nM T67162 D0B1GJ 44578927 Ki > 10000 nM T67162 D0B9DR 15508243 Ki = 5300 nM T67162 D0C0UM 10775317 Ki > 20000 nM T67162 D0C5RZ 5610 Ki > 17000 nM T67162 D0C7SE 16756754 Ki = 7400 nM T67162 D0CA9H 25107518 Ki = 503 nM T67162 D0D3YN 1238 Ki = 0.67 nM T67162 D0E1PL 9865384 Ki = 15000 nM T67162 D0E1RX 11335419 Ki = 1006 nM T67162 D0E3AL 56597938 Ki = 0.2 nM T67162 D0F0IA 11301655 Ki > 6000 nM T67162 D0F6CD 5202 IC50 = 0.0003 nM T67162 D0FF6S 16038374 IC50 > 10000 nM T67162 D0FL1D 9842124 Ki = 1600 nM T67162 D0FU2V 24754478 Ki = 26 nM T67162 D0FU5E 10220053 Ki > 1000 nM T67162 D0G0IQ 3802 Ki = 5940 nM T67162 D0G2CP 10404144 Ki = 2200 nM T67162 D0G2HT 22397829 Ki = 392 nM T67162 D0G7LE 10991121 Ki > 1500 nM T67162 D0G8CV 9954003 Ki = 0.7943 nM T67162 D0G8VU 3645619 Ki = 1100 nM T67162 D0H2IT 9928335 Ki = 2748 nM T67162 D0H2WQ 54562 EC50 = 1.2 nM T67162 D0H3KU 172267 Ki = 6 nM T67162 D0H7PC 6918553 Ki > 5011.87 nM T67162 D0H9QG 5312148 Ki = 3981 nM T67162 D0HG4U 11515697 Ki = 88 nM T67162 D0I2WQ 44579031 Ki > 10000 nM T67162 D0I9KV 11220599 IC50 > 10000 nM T67162 D0IU8V 9903877 Ki = 4.25 nM T67162 D0J1HP 10378389 EC50 = 0.01995 nM T67162 D0K3UL 9796720 Ki = 120 nM T67162 D0L3XU 122187 Ki = 3760 nM T67162 D0L5MW 181743 Ki = 858 nM T67162 D0L7OM 6917970 Ki = 11 nM T67162 D0L7ZD 56593482 Ki = 1.2 nM T67162 D0LR8X 1243 Ki = 1360 nM T67162 D0LV7U 10667433 Ki = 286 nM T67162 D0M2BB 25333445 Ki = 2400 nM T67162 D0M2ZE 6604756 Ki = 13 nM T67162 D0M3PV 133633 Ki = 2.4 nM T67162 D0M5XV 24866114 EC50 = 13.4 nM T67162 D0M5ZE 5311416 Ki = 316.23 nM T67162 D0M7SY 9910352 Ki = 100 nM T67162 D0M8LN 9806160 Ki = 320 nM T67162 D0N6OL 11452268 IC50 > 100000 nM T67162 D0ND5D 10493741 Ki > 1700 nM T67162 D0O1PM 4420454 Ki = 34 nM T67162 D0O3GF 1220 Ki = 84 nM T67162 D0O4BC 11776546 Ki = 75.8 nM T67162 D0O7DA 37459 Ki = 0.04 nM T67162 D0O9BZ 2728532 Ki = 53 nM T67162 D0OG0R 10337743 IC50 < 5000 nM T67162 D0P0IX 16104 IC50 = 34 nM T67162 D0P4BY 146265 Ki = 1374 nM T67162 D0P7OB 9798466 Ki = 5882 nM T67162 D0PV6G 115007 Ki = 251.19 nM T67162 D0Q2GP 10381810 Ki = 150 nM T67162 D0Q2MX 56599142 EC50 = 50 nM T67162 D0Q4DP 6603897 Ki > 1700 nM T67162 D0Q5IP 10851078 Ki = 110 nM T67162 D0Q7FM 15443 Ki = 52 nM T67162 D0R3GW 10296414 Ki = 1258.93 nM T67162 D0R5QM 10354670 Ki = 20.6 nM T67162 D0R5WB 9817960 Ki = 896 nM T67162 D0R8PL 44579030 Ki > 10000 nM T67162 D0R8UU 44396220 Ki = 1015 nM T67162 D0RC9T 9795587 Ki > 1300 nM T67162 D0RQ8R 11973809 Ki = 5000 nM T67162 D0S1XN 44323962 Ki = 47 nM T67162 D0SL4Q 46190878 Ki > 10000 nM T67162 D0T1TU 68950 Ki = 2024 nM T67162 D0T2RY 9948320 Ki = 77 nM T67162 D0T3IH 119146 Ki = 0.133 nM T67162 D0TU5W 44323978 Ki = 81.3 nM T67162 D0U0VH 9904242 Ki = 35 nM T67162 D0V4NW 25139332 Ki = 8800 nM T67162 D0V4RP 1346 Ki = 679.6 nM T67162 D0V5OY 16725912 Ki > 1000 nM T67162 D0V5SQ 68186 Ki = 3 nM T67162 D0WD6J 10357869 Ki = 320 nM T67162 D0WU9R 133008 Ki > 1700 nM T67162 D0X1QW 122334 Ki = 14 nM T67162 D0X2NO 3153 IC50 = 0.00000004 nM T67162 D0X3JB 11529282 Ki = 664 nM T67162 D0X4PH 11224758 Ki = 7.3 nM T67162 D0X5LJ 12988959 Ki = 349 nM T67162 D0X8LG 11243002 IC50 > 10000 nM T67162 D0Z1OF 23643664 Ki = 224 nM T97903 D00SQN 12136798 IC50 = 760 nM T97903 D0E3SH 6918837 IC50 = 1.6 nM T97903 D0E7PQ 5311 Ki = 13 nM T97903 D0L7LC 5352062 IC50 = 0.3 nM T97903 D00FHR 9865515 IC50 = 590 nM T97903 D05KED 53340666 IC50 > 10000 nM T97903 D07FPY 6918877 Ki = 12.8 nM T97903 D09XIZ 11538455 Ki = 0.07 nM T97903 D0B3FV 6445533 IC50 = 5.58 nM T97903 D0E6UZ 54575456 IC50 = 132 nM T97903 D0L2UQ 49855250 Ki = 43 nM T97903 D0M8FD 4261 IC50 = 900 nM T97903 D0XT6W 6918638 Ki = 27 nM T97903 D0J8OC 5186 IC50 = 5200 nM T97903 D00HXJ 118884610 Ki = 495 nM T97903 D0N2DK 72710871 IC50 = 55.5 nM T97903 D0QX3G 71532921 IC50 > 10000 nM T97903 D0ZG5X 71811260 IC50 = 656 nM T97903 C18ENP 6918846 Ki = 14 nM T97903 CC0EU7 9828788 IC50 = 2360 nM T97903 C7RC1E 10309899 IC50 = 2.1 nM T97903 C8G5WP 11210533 IC50 = 12900 nM T97903 CG9OC4 11682502 IC50 = 20.7 nM T97903 CYB26W 11688197 IC50 > 1000 nM T97903 CE4Z0Y 11844891 IC50 = 30700 nM T97903 C0QCW4 11988293 IC50 = 77000 nM T97903 C9G1BN 11993595 IC50 = 410 nM T97903 C2D1KP 15983982 Ki = 11 nM T97903 CHB82E 15986417 IC50 = 57200 nM T97903 C52EVH 15986418 IC50 = 5010 nM T97903 CS1QO9 15986509 IC50 = 73000 nM T97903 CFK8J5 16068056 Ki = 14 nM T97903 CMQP70 16068495 Ki = 18 nM T97903 CT84XO 16068594 Ki = 14 nM T97903 CF3ZG5 16068595 Ki = 13 nM T97903 CL60CA 16068912 Ki = 4.2 nM T97903 C9ZQB3 16095102 Ki > 5000 nM T97903 C80XYC 16095113 Ki > 5000 nM T97903 CWO7V0 16733295 IC50 = 190 nM T97903 CV54SY 16733414 IC50 = 610 nM T97903 C8RC9P 24744325 IC50 = 25000 nM T97903 C17GDO 24779722 IC50 = 197 nM T97903 CX69SY 25066355 IC50 = 1210 nM T97903 CF8VP4 25066356 IC50 = 564 nM T97903 CS9XH7 25066547 IC50 = 546 nM T97903 C46AGN 25066548 IC50 = 57.7 nM T97903 CJF2M7 25066549 IC50 = 226 nM T97903 CCD5M7 25227504 IC50 = 22.9 nM T97903 CK0D5S 25227505 IC50 = 97.1 nM T97903 CN97JP 25227508 IC50 = 103 nM T97903 CW8R1B 25227513 IC50 = 174 nM T97903 C43BHY 25269097 IC50 = 37000 nM T97903 CJ1RQ7 42598706 IC50 = 1130 nM T97903 C1UAO7 42601485 IC50 > 50000 nM T97903 CDT65Y 42631047 IC50 > 100000 nM T97903 CO57GS 44138033 IC50 = 10800 nM T97903 C86IOC 44328927 IC50 = 9350 nM T97903 C5VP4D 44454144 IC50 > 50000 nM T97903 CIO34V 44564642 Ki = 16 nM T97903 CA6Q9Y 44592060 IC50 = 6260 nM T97903 C5H8RA 44598536 IC50 = 300 nM T97903 C42SJP 45141750 IC50 = 1600 nM T97903 CLE9U5 45141751 IC50 = 78.6 nM T97903 CSM1O6 45271073 IC50 = 5800 nM T97903 CQ69AM 46205433 IC50 = 75.1 nM T97903 CPSI47 46890583 Ki = 9 nM T97903 C90NYX 46896338 IC50 = 14000 nM T97903 CL7PS1 49831258 IC50 > 50000 nM T97903 CI5L2P 49846123 IC50 = 160.87 nM T97903 C4DL0M 49847150 IC50 = 54.7 nM T97903 CC7Y9U 49850262 IC50 > 30000 nM T97903 C50PXU 49855444 IC50 > 50000 nM T97903 C78GKN 53361474 IC50 = 476 nM T97903 CNB63X 53361475 IC50 = 116 nM T97903 CQ43VH 53363518 Ki = 8.8 nM T97903 C6Y2EV 53374826 IC50 = 5530 nM T97903 C5A7MU 54613496 IC50 = 33.4 nM T97903 C7R9TZ 56663191 IC50 = 3 nM T97903 CZ25SN 56935695 IC50 > 30000 nM T97903 CA5Q6O 58147189 IC50 > 50000 nM T97903 C4DYC0 58147224 IC50 > 50000 nM T97903 CMP04X 58147302 IC50 > 50000 nM T97903 CLD40J 58465708 IC50 = 29000 nM T97903 C1MB4Q 59323957 IC50 > 30000 nM T97903 CK6LX0 59454220 IC50 > 30000 nM T97903 C2SDN1 59454252 IC50 = 20000 nM T97903 CB7X2E 60151224 IC50 > 10000 nM T97903 CY05OU 60151225 IC50 > 10000 nM T97903 CWO8H0 60152596 IC50 > 10000 nM T97903 CBN3L0 69950064 Ki > 19000 nM T97903 C6RFQ8 70676597 IC50 > 20000 nM T97903 CQY1I6 70789579 Ki > 19000 nM T97903 C0LWJ6 71520631 IC50 = 2135 nM T97903 CO28HI 71520716 IC50 = 997 nM T97903 CVA5Q7 71520717 IC50 = 852 nM T97903 C6KBD4 71534512 IC50 = 24 nM T97903 CT51EW 71534810 IC50 = 3 nM T97903 C7QN3O 71534812 IC50 = 1 nM T97903 C8M3HU 71537640 IC50 = 12 nM T97903 C2QML7 71537641 IC50 = 4 nM T97903 CZJX53 71537927 IC50 = 293 nM T97903 CU0ZE6 71537928 IC50 = 14 nM T97903 CH9FS7 71537929 IC50 = 82 nM T97903 CTW95A 71537931 IC50 = 15 nM T97903 CW3BT5 71537932 IC50 = 14200 nM T97903 C3C0RO 71538475 IC50 = 5 nM T97903 CIA28E 71538746 IC50 = 6 nM T97903 CFCV26 71538748 IC50 = 293 nM T97903 CY2T1Q 71538749 IC50 = 140 nM T97903 C4A6VJ 71538750 IC50 = 10 nM T97903 CG72NC 71538751 IC50 = 13 nM T97903 CKR6U8 71583101 IC50 = 9700 nM T97903 C0P8CH 71748076 IC50 = 1320 nM T97903 CTSK68 71811225 IC50 = 4080 nM T97903 C1K6OW 71811226 IC50 = 2440 nM T97903 CU3N9R 71811227 IC50 = 1350 nM T97903 CS2L4B 71811228 IC50 = 1210 nM T97903 CL4DT9 71811229 IC50 = 730 nM T97903 CK6DB4 71811230 IC50 = 5590 nM T97903 CHR8V0 71811259 IC50 = 2950 nM T97903 CVL54T 71811261 IC50 = 37100 nM T97903 CZR93K 71811262 IC50 = 4250 nM T97903 CM8BE4 71811290 IC50 = 3910 nM T97903 C0MV3O 71811291 IC50 > 10000 nM T97903 C7UYD4 71811292 IC50 = 5220 nM T97903 C7XL3N 71811293 IC50 > 10000 nM T97903 C4HBC5 71811294 IC50 = 3740 nM T97903 CTA26S 71811295 IC50 = 4680 nM T97903 CI9H6L 72164895 IC50 = 224 nM T97903 CS5UL7 72195322 IC50 = 2342 nM T97903 CV09DJ 72734543 IC50 = 5000 nM T97903 CS6LW0 72946640 IC50 = 47 nM T97903 CXM37Z 72946641 IC50 = 75 nM T97903 CQA16N 72946833 IC50 = 13 nM T97903 CNR7Z2 72946834 IC50 = 255 nM T97903 C12JYS 72946835 IC50 = 150 nM T97903 C5Y9XH 72946836 IC50 = 70 nM T97903 CVZR94 72946837 IC50 = 1440 nM T97903 C8-AUG 72946838 IC50 = 262 nM T97903 CHQ39Y 72947043 IC50 = 135 nM T97903 CCST90 72947044 IC50 = 15 nM T97903 C7J3RH 72947045 IC50 = 127 nM T97903 CK10LZ 73292342 IC50 > 30000 nM T97903 CZB6G7 73776472 IC50 = 900.4 nM T97903 C3UC9H 73891099 IC50 = 11700 nM T97903 CL4JQ3 76331862 IC50 = 2630 nM T97903 C08CPW 76335428 IC50 = 47.8 nM T97903 C06YBD 86302594 IC50 = 521 nM T97903 CS5I4Y 87261507 IC50 = 340 nM T97903 CB47VC 89464167 IC50 = 949 nM T97903 CYW51P 90654946 IC50 = 63400 nM T97903 CJH1S6 90654947 IC50 = 38100 nM T97903 CSR56C 90655296 IC50 = 1770 nM T97903 CSDO81 90664458 Ki = 24 nM T97903 CJO6T1 91810840 IC50 = 3700 nM T97903 CYJ12Q 91884636 IC50 = 14 nM T97903 C34WIG 92045024 IC50 > 100000 nM T97903 C9OC0F 101882265 IC50 = 75300 nM T97903 C2I8XR 101882814 Ki = 6000 nM T97903 C8KZB4 101883993 Ki = 1500 nM T97903 C7Q6ID 101884982 IC50 = 30 nM T97903 CR46PQ 101884983 IC50 = 10 nM T97903 CRZ83C 101884989 IC50 = 102 nM T97903 CT7Z8F 102514716 IC50 = 32820 nM T97903 CSU52M 118656852 IC50 = 500 nM T97903 CB6AJ9 118656853 IC50 = 17000 nM T97903 C45UYG 118709095 IC50 = 74000 nM T97903 C7QHE4 118712502 IC50 = 0.1 nM T97903 C8KSD6 118712503 IC50 = 0.2 nM T97903 CXF0U3 118714375 IC50 = 897 nM T97903 CY4GN9 118714377 IC50 = 1725 nM T97903 CM5QT7 118719376 Ki = 3200 nM T97903 CPB7C3 118719377 Ki = 1300 nM T97903 C09OGH 118719378 Ki = 1100 nM T97903 CR5VC1 118719379 Ki = 2000 nM T97903 C32LCM 118719380 Ki = 1000 nM T97903 C8U6YR 118719381 Ki = 300 nM T97903 C9Y0HV 118719382 Ki = 800 nM T97903 CY0J4D 118719383 Ki = 900 nM T97903 CCYU59 118719817 IC50 = 44 nM T97903 CUI51W 118720529 IC50 = 52.7 nM T97903 CMV2W9 118721625 IC50 = 9 nM T97903 CF5TO3 118721859 IC50 = 67 nM T97903 CK97TZ 118721860 IC50 = 62 nM T97903 CYV30O 118721861 IC50 = 5 nM T97903 C5WYI1 118721862 IC50 = 12 nM T97903 CSMW25 118721863 IC50 = 776 nM T97903 C5B1KM 118721864 IC50 = 89 nM T97903 CG8LZ0 118721865 IC50 = 2070 nM T97903 CPCN23 118721866 IC50 = 1840 nM T97903 CM0A9U 118721867 IC50 = 1870 nM T97903 CI8G4X 118737400 IC50 = 10200 nM T97903 C2F8TQ 118737455 IC50 = 608 nM T97903 CIA40K 121472983 IC50 = 15000 nM T97903 C28JVO 122192004 IC50 > 10000 nM T97903 CF2D8U 122192005 IC50 > 10000 nM T97903 C5W8OZ 122376192 IC50 = 290 nM T97903 C3V5ND 122550211 IC50 > 10000 nM T97903 CZE35C 122648343 IC50 > 10000 nM T97903 C54RNT 122648367 IC50 > 1000 nM T97903 C1UVI7 122648600 IC50 > 1000 nM T97903 CMX59K 122648648 IC50 > 1000 nM T97903 CVZ64I 122648649 IC50 = 835 nM T97903 CE4CI8 127025178 IC50 > 10000 nM T97903 CG8NU7 127027995 IC50 > 10000 nM T97903 CV07OM 127028943 IC50 > 10000 nM T97903 CV9I8D 127030313 IC50 = 16200 nM T97903 CA9EV6 130205513 IC50 = 5000 nM T97903 C8KRX0 130205516 IC50 = 10000 nM T97903 CJ7CQ5 130205526 IC50 = 8000 nM T97903 CMZ6B2 130226783 IC50 = 11000 nM T97903 C6OXE3 132134663 IC50 = 930 nM T97903 C6X3HG 132145728 IC50 = 1004 nM T97903 C8O9DP 132157820 IC50 = 376 nM T97903 C4KE3N 132938351 IC50 > 10000 nM T97903 CH4TU5 134492521 IC50 = 2 nM T97903 C05FVT 134492522 IC50 = 3 nM T97903 C14FWK 135348858 IC50 = 5120 nM T97903 C95PIU 136048746 IC50 = 1200 nM T97903 CT19ND 136110961 IC50 > 100000 nM T97903 CY9U0E 136173089 IC50 = 100 nM T97903 C67EFJ 137628684 IC50 > 1000 nM T97903 CX0PH5 137628685 IC50 = 636 nM T97903 C6JVG9 137635398 IC50 = 31 nM T97903 CJF39U 137644905 IC50 = 2140 nM T97903 C8GNS5 137645287 IC50 = 8870 nM T97903 C5FHD3 137652442 IC50 = 12900 nM T97903 C1SBN5 137654946 IC50 = 651 nM T97903 C76OGQ 137656942 IC50 = 2400 nM T97903 CAQ62X 137701235 Ki = 21 nM T97903 CVA12U 138377601 IC50 = 13900 nM T97903 CA3C4O 138454792 IC50 > 1000 nM T97903 CN2UH1 139303146 IC50 = 77.82 nM T97903 C7XI0V 141764754 IC50 > 10000 nM T97903 CX0E9B 142505968 IC50 = 9819 nM T97903 C9G5ZW 142505990 IC50 = 9000 nM T97903 CBJC50 142505992 IC50 = 23030 nM T97903 C7N8LV 142506025 IC50 = 3362 nM T97903 CKBF56 142506033 IC50 = 2089 nM T97903 CLND62 142506170 IC50 = 74140 nM T97903 CGNQ74 142506189 IC50 = 324 nM T97903 C1T3IQ 142506210 IC50 = 2155 nM T97903 CEGV67 142506220 IC50 = 1778 nM T97903 CKG98W 145953085 IC50 > 10000 nM T97903 CUX8C2 145960671 IC50 = 85 nM T97903 CE3T9X 145960682 IC50 > 10000 nM T97903 C0FI2X 145960809 IC50 = 300 nM T97903 CK1XI0 145960971 IC50 > 10000 nM T97903 CT3WX0 145961194 IC50 = 1 nM T97903 C7IUK3 145961289 IC50 = 3 nM T97903 C5OI0Y 145961494 IC50 = 170 nM T97903 CJOL50 145961514 IC50 = 2 nM T97903 C0PSA7 145961516 IC50 = 2300 nM T97903 CB9G4Q 145961803 IC50 = 2100 nM T97903 C12XQF 145961873 IC50 = 4600 nM T97903 CYHO80 145962011 IC50 = 6 nM T97903 CZ1V7L 145962017 IC50 = 26 nM T97903 CSRO14 145962110 IC50 = 27 nM T97903 CU3E7A 145962221 IC50 = 7 nM T97903 C2X5WR 145962427 IC50 = 2 nM T97903 CRZ1M3 145962635 IC50 = 30 nM T97903 CDR1E6 145962762 IC50 = 1200 nM T97903 CR7H8C 145963476 IC50 = 7 nM T97903 C40QIR 145963557 IC50 = 35 nM T97903 CX0OD9 145968046 IC50 = 76.3 nM T97903 C2XS8E 145968675 IC50 = 3500 nM T97903 CUI37A 145969799 IC50 = 175.9 nM T97903 CWD0A9 145983712 Ki = 140 nM T97903 C56MWZ 145986208 Ki = 38 nM T97903 C7L1GU 145986811 IC50 = 15.8 nM T97903 C0GMR1 146585718 IC50 = 2255 nM T97903 C0YXS8 147254231 IC50 = 80020 nM T97903 CN71OS 149405396 IC50 > 100000 nM T97903 CH3JE4 150054712 IC50 = 14730 nM T97903 C8S3MF 150076000 IC50 > 300 nM T97903 CU2XY0 150312795 IC50 = 10500 nM T97903 C5PQI9 150470306 IC50 = 25050 nM T97903 C4JP7X 150533939 IC50 = 5501 nM T97903 C89BKD 150622000 IC50 > 10000 nM T97903 CIM06Z 150916115 IC50 = 7392 nM T97903 CM6IF7 151532669 IC50 = 11290 nM T97903 CS0V6U 151543423 IC50 = 16740 nM T97903 CV39LB 151825687 IC50 > 10000 nM T97903 CROU95 152148008 IC50 = 5686 nM T97903 CY1NG0 152157103 IC50 = 52050 nM T97903 CYF2I5 152375216 IC50 = 19800 nM T97903 CL1UA7 152547478 IC50 = 15400 nM T97903 C2AOQ6 152562172 IC50 = 10660 nM T97903 CT4H9P 153408403 IC50 = 34370 nM T97903 CK7P3F 153408410 IC50 = 13850 nM T97903 C9FIY4 153534005 IC50 > 10000 nM T97903 CPF6R7 155512997 IC50 > 1000 nM T97903 CA1J3N 155517086 IC50 > 100000 nM T97903 CY54TU 155518062 IC50 = 17000 nM T97903 CEH2N5 155518106 IC50 > 100000 nM T97903 C41AIO 155518963 IC50 = 346 nM T97903 CAD06U 155519254 IC50 = 1050 nM T97903 CDY5H6 155519645 IC50 = 1890 nM T97903 CAZ3S7 155521187 IC50 = 820 nM T97903 CZ75FW 155521272 IC50 > 100000 nM T97903 CQ4RG3 155528629 IC50 = 210 nM T97903 C9L6OC 155529247 IC50 > 1000 nM T97903 COTR30 155530602 IC50 > 1000 nM T97903 C47WTL 155531016 IC50 = 1020 nM T97903 CIZ46A 155533876 IC50 = 540 nM T97903 C6LB5D 155535084 IC50 = 1500 nM T97903 CJH9L4 155535498 IC50 > 1000 nM T97903 CTF98X 155537473 IC50 = 80 nM T97903 C63FKN 155538445 IC50 = 8120 nM T97903 CLD19W 155539311 IC50 = 3610 nM T97903 CKZ9A5 155543845 IC50 > 1000 nM T97903 CJK31W 155544599 IC50 = 190 nM T97903 C1VF5A 155544728 IC50 > 1000 nM T97903 CS3GO2 155546558 IC50 = 150 nM T97903 CCTU12 155549163 IC50 = 254 nM T97903 CEO4J8 155551917 IC50 = 1577 nM T97903 C46WHP 155552329 IC50 = 253 nM T97903 CGDF76 155554360 IC50 = 2400 nM T97903 CIN57Q 155556138 IC50 = 1810 nM T97903 CJ9FW6 155557777 IC50 = 837 nM T97903 CJ3MZ1 155558467 IC50 = 665 nM T97903 C8AUB0 155558567 IC50 = 632 nM T97903 C0RZ7V 155558710 IC50 = 304 nM T97903 C2IS1E 155559200 IC50 = 3229 nM T97903 C28CVZ 155559279 IC50 = 51.9 nM T97903 CPD50Q 155559583 IC50 = 6600 nM T97903 CY3XI1 155559600 IC50 = 191 nM T97903 CMD6Q7 155560250 IC50 = 1220 nM T97903 C9UYZ6 155564157 IC50 = 1365 nM T97903 C4IM1X 155564305 IC50 = 697 nM T97903 CE0U7K 155564881 IC50 = 396 nM T97903 CZDC03 155565491 IC50 = 1200 nM T97903 C3G1JV 155565712 IC50 = 288 nM T97903 CT6Z4H 155567814 IC50 = 3164 nM T97903 C5NQK8 155569352 IC50 = 3962 nM T97903 D00GBB 11449246 Ki = 39 nM T97903 D00SEE 11379392 IC50 = 262 nM T97903 D01YBR 44591988 IC50 = 3060 nM T97903 D04KQF 6675804 Ki = 718.7 nM T97903 D04UVL 1133083 IC50 > 50000 nM T97903 D05OVV 11993691 IC50 = 430 nM T97903 D09RKA 72946782 IC50 = 5000 nM T97903 D0B3ZM 11436024 IC50 = 659 nM T97903 D0E0TA 44454650 IC50 > 50000 nM T97903 D0E9DD 16095101 Ki = 60 nM T97903 D0M1ZI 16095112 Ki > 5000 nM T97903 D0M9LJ 44454415 IC50 > 50000 nM T97903 D0MD7H 44454143 IC50 > 50000 nM T97903 D0N9AK 44138031 IC50 = 5480 nM T97903 D0Q2GM 44454416 IC50 > 50000 nM T97903 D0Q5DI 71462653 IC50 = 5140 nM T97903 D0Q9PO 16095114 Ki = 35 nM T97903 D0T0SK 44138032 IC50 = 790 nM T97903 D0U8FC 759408 IC50 > 50000 nM T97903 D0XZ9Q 11149404 IC50 = 133 nM T97903 D0Z8PX 24757913 IC50 > 10000 nM T82795 C0M5JG 360901 Ki = 5900 nM T82795 C8ESO9 541913 Ki > 2000000 nM T82795 CE0OX8 568763 Ki = 310000 nM T82795 CI3E4C 673949 Ki = 1700000 nM T82795 CQ3U6R 684781 Ki = 120000 nM T82795 C40SXF 689303 Ki = 240000 nM T82795 CQK9D6 723206 Ki = 1700000 nM T82795 C63XJQ 1416323 Ki = 80000 nM T82795 CV5XG6 1749091 Ki = 1200 nM T82795 CK5D2F 1896476 Ki = 13000 nM T82795 CB9QX6 2195375 Ki = 8800 nM T82795 CAH80O 4417218 Ki > 2000000 nM T82795 CK0PN6 5967294 Ki = 54000 nM T82795 C42KNA 6622273 Ki = 370000 nM T82795 CH7CE6 9836739 Ki = 1800 nM T82795 CDQ43L 10930781 IC50 < 10000 nM T82795 C2DG9Y 71625260 Ki = 21000 nM T82795 C4XLD5 71695771 Ki = 3100 nM T82795 C82GTD 73348987 IC50 < 10000 nM T82795 CQUW87 73353527 IC50 < 10000 nM T82795 CV82OR 90656496 Ki = 1300 nM T82795 C8RX0F 122180635 Ki = 2700 nM T82795 C13NQI 122180636 Ki = 63000 nM T82795 CYS9P7 122180637 Ki = 4100 nM T82795 CI58UX 122180638 Ki > 100000 nM T82795 CG69NB 122180639 Ki = 3300 nM T82795 C7MW3Q 122180640 Ki = 52000 nM T82795 CZE8K1 122180708 Ki = 1000 nM T82795 CC5OM8 122180709 Ki > 130000 nM T82795 C3JB7G 122180710 Ki = 39000 nM T82795 C9HB0D 122180711 Ki = 120000 nM T82795 CJY3B8 122180712 Ki = 17000 nM T82795 C7GHX0 122180713 Ki = 51000 nM T82795 CCU3P8 135475052 Ki = 8700 nM T82795 CZ41FV 135995896 Ki = 230000 nM T82795 CF3WR1 146670445 Ki = 6700 nM T82795 CB8LK7 146671571 Ki = 2900 nM T82795 C39ETG 146671572 Ki = 10000 nM T82795 CP49XD 155512566 Ki = 8500 nM T82795 CN35MG 155512758 Ki = 8000 nM T82795 C7WI9H 155513400 Ki = 70000 nM T82795 C63ZDX 155514892 Ki = 14000 nM T82795 C7VN0G 155514942 Ki > 100000 nM T82795 C53IGM 155516253 Ki = 25000 nM T82795 CSP78U 155518565 Ki > 100000 nM T82795 C01BIC 155518610 Ki = 7600 nM T82795 C0Q6YO 155520646 Ki = 2200 nM T82795 C57CGM 155520694 Ki = 89000 nM T82795 C7SC2F 155522080 Ki = 3700 nM T82795 CV9WD0 155522143 Ki = 640 nM T82795 C79WQC 155522343 Ki = 1900 nM T82795 C1MNV7 155522353 Ki > 100000 nM T82795 CM51NC 155522369 Ki = 17000 nM T82795 COM6S5 155523009 Ki = 9700 nM T82795 CQGZ01 155524335 Ki = 3100 nM T82795 CY78QE 155524414 Ki = 22000 nM T82795 CS2Y6J 155524482 Ki = 2600 nM T82795 CY8M3N 155524656 Ki = 20000 nM T82795 CY2V3K 155527310 Ki = 2500 nM T82795 CW19AX 155527817 Ki > 100000 nM T82795 C1ZIE9 155529701 Ki > 100000 nM T82795 C4P9BZ 155529836 Ki = 1500 nM T82795 CEA1Q4 155529863 Ki = 16000 nM T82795 C1BGD3 155530410 Ki = 1900 nM T82795 C8WY6N 155530942 Ki = 3300 nM T82795 C6N0VR 155531142 Ki = 5200 nM T82795 CX83AR 155533295 Ki = 11000 nM T82795 C5QA0O 155534911 Ki = 9300 nM T82795 C6R1DA 155535578 Ki = 8900 nM T82795 CK12FM 155538511 Ki > 100000 nM T82795 CB51VK 155539480 Ki = 2300 nM T82795 CAXD47 155539905 Ki = 3600 nM T82795 CT62XE 155545293 Ki = 2600 nM T82795 CNA7Z3 155545420 Ki = 440 nM T82795 CMH32L 155545837 Ki > 100000 nM T82795 CE8AQ9 155547268 Ki = 2700 nM T82795 C6XR8G 155547949 Ki = 3300 nM T82795 C5URK8 155549143 Ki = 3300 nM T82795 CW1E8U 155551766 Ki = 15000 nM T82795 C0BZ8G 155553111 Ki = 4300 nM T82795 CTL90A 155555958 Ki = 11000 nM T82795 C71TKZ 155556130 Ki = 15000 nM T82795 C3J7KU 155556445 Ki > 100000 nM T82795 CWU7M0 155558775 Ki = 9600 nM T82795 C23BPR 155559087 Ki = 3900 nM T82795 CA9H7Z 155561933 Ki > 100000 nM T82795 CAY09N 155562046 Ki = 10000 nM T82795 C4V9EC 155564679 Ki = 4900 nM T82795 CR20HP 155565262 Ki = 2400 nM T82795 CS62JP 155567741 Ki = 6600 nM T82795 C1FQ9T 155567749 Ki = 12000 nM T82795 CRD5F9 155568218 Ki = 4500 nM T82795 D07WDQ 66541 Ki = 3800 nM T82795 D0L7DB 482190 IC50 < 10000 nM T30727 D0J3SU 9847835 Ki > 5000 nM T30727 CV7IN2 104934 Ki = 337 nM T30727 C1KR5B 5327301 Ki = 96000 nM T30727 C37TKL 5327302 Ki = 21000 nM T30727 C64ZMN 5327304 Ki = 92000 nM T30727 C3IZ2W 5327307 Ki = 13000 nM T30727 C16DTL 5327308 Ki = 38000 nM T30727 C4O3QY 5327309 Ki > 100000 nM T30727 C3GUM7 5327310 Ki = 27000 nM T30727 CFN2P6 9800285 Ki = 30000 nM T30727 C4XO3K 9821545 Ki = 33000 nM T30727 CLAC59 9828058 Ki = 248 nM T30727 C6S3KT 9840223 Ki > 25000 nM T30727 CX67SZ 10826725 Ki = 5000 nM T30727 CDX7A4 10963183 Ki = 22000 nM T30727 CDT9G3 11467504 IC50 = 0.5 nM T30727 CJ57OA 14585243 Ki = 207 nM T30727 C25ELB 44143088 IC50 = 33113.11 nM T30727 CD8WB9 44304162 Ki > 50000 nM T30727 C8D5TB 44364680 Ki = 38000 nM T30727 C86ORE 44459987 IC50 = 8128.31 nM T30727 CDY2W5 49796910 IC50 = 0.3 nM T30727 CGY3W2 71471109 IC50 = 510 nM T30727 CANH70 71716242 IC50 = 5600 nM T30727 C40WIR 71718085 IC50 = 180 nM T30727 CU75VK 71719897 IC50 = 370 nM T30727 CBV6F1 71720507 IC50 = 90 nM T30727 CID3N6 134134572 IC50 > 5000 nM T30727 CV0R3B 134135432 Ki = 267 nM T30727 C3D7LQ 134136688 Ki = 870 nM T30727 CBY95D 134138690 IC50 > 5000 nM T30727 CG3EI1 134145896 Ki = 148 nM T30727 CI9X3K 134147411 Ki = 8 nM T30727 CP16IA 134148745 Ki = 276 nM T30727 CPE90G 134149983 Ki = 393 nM T30727 CBE39C 134151245 Ki = 563 nM T30727 CY0LD4 134152014 Ki = 306 nM T30727 C3K5HR 134153309 Ki = 119 nM T30727 CWQT79 134156687 Ki = 215 nM T30727 D0N5MU 4117381 Ki > 50000 nM T30727 D0Q9XX 515950 Ki = 4000 nM T30727 D0Y5IQ 44255320 IC50 = 5000 nM T00075 D0E3TC 44259 IC50 = 5.35 nM T00075 CBOP58 11293798 Ki = 6630 nM T00075 C26BZX 11362471 Ki = 4440 nM T00075 CWXB93 11397177 Ki > 10000 nM T00075 C7YG1N 24759534 IC50 = 1200 nM T00075 CCK8D2 25154767 IC50 = 210 nM T00075 C7BAN0 25262260 IC50 = 150 nM T00075 CR7TY6 44197572 IC50 = 5350 nM T00075 C1G2ZQ 44198874 IC50 = 333 nM T00075 CKV96M 44571730 IC50 = 79 nM T00075 CG6UW5 44634494 IC50 = 247 nM T00075 CA4XQ3 45375859 IC50 = 9552 nM T00075 CLS29B 46872626 IC50 > 10000 nM T00075 CQIC19 46879806 IC50 = 7861 nM T00075 C2O8RZ 46886323 IC50 > 1000 nM T00075 CA2Y8J 46901260 IC50 = 810 nM T00075 CXJ63M 59603829 IC50 = 9200 nM T00075 CQEU96 59603842 IC50 = 72 nM T00075 CC7A5F 66577033 IC50 = 127 nM T00075 CV63UL 67240318 IC50 > 10000 nM T00075 C69OHY 68560854 IC50 = 4306 nM T00075 CCD89X 68563058 IC50 = 8695 nM T00075 CW6BH7 68566254 IC50 = 6400 nM T00075 C48EIQ 68568011 IC50 = 1853 nM T00075 CAWC35 68621678 IC50 > 1000 nM T00075 C5DGR9 69036886 IC50 = 10000 nM T00075 C8AM1K 71655603 IC50 = 1550 nM T00075 C0DL3F 72698602 IC50 = 2.87 nM T00075 C1HW4B 89735655 IC50 = 1000 nM T00075 COA09T 90668074 IC50 = 8640 nM T00075 CEN9Z0 90668075 IC50 = 1275 nM T00075 C9JW0N 90668076 IC50 > 20000 nM T00075 COX43L 90668077 IC50 = 261 nM T00075 CL56TZ 90668078 IC50 > 20000 nM T00075 C7Z6AG 90668079 IC50 = 294 nM T00075 CIT61M 90668081 IC50 = 74 nM T00075 CM2UH4 135894362 IC50 > 1000 nM T00075 CY19DW 135894364 IC50 > 1000 nM T00075 C15HQK 136218656 IC50 > 1000 nM T00075 CZ06UK 136218660 IC50 > 1000 nM T00075 CML48X 136218661 IC50 > 1000 nM T00075 COB69I 136218662 IC50 > 1000 nM T00075 CSL6Q8 136218663 IC50 > 1000 nM T00075 CTFJ83 136226213 IC50 > 1000 nM T00075 C5EV8A 136240902 IC50 > 1000 nM T00075 CX9LB5 136240903 IC50 > 1000 nM T00075 CMC58H 136240944 IC50 > 1000 nM T00075 C60PRZ 136241012 IC50 > 1000 nM T00075 C1Q9YN 136252259 IC50 > 1000 nM T00075 C2MD1Q 155513187 IC50 > 10000 nM T00075 D00ERW 44444843 Ki > 9524 nM T00075 D0R3MO 46864283 IC50 = 669 nM T02446 D03LWG 53235510 IC50 = 3039 nM T02446 D0E3TC 44259 IC50 = 60.3 nM T02446 D03BNU 59604787 IC50 > 10000 nM T02446 D0T3ME 156422 IC50 = 110 nM T02446 CQN3Z7 24825710 IC50 = 1110 nM T02446 CY8L7E 24896769 IC50 > 10000 nM T02446 C2ICS7 25065806 IC50 = 6 nM T02446 C0SWH5 53348216 IC50 > 40000 nM T02446 C8NA4L 53384644 IC50 > 30000 nM T02446 CK6WO0 66552478 IC50 < 10000 nM T02446 CV63UL 67240318 IC50 > 10000 nM T02446 CQC0R5 68181954 IC50 > 10000 nM T02446 CPG3A5 86302574 IC50 > 30000 nM T02446 C9WGB8 127035904 IC50 = 2500 nM T02446 CUO0C5 132156633 IC50 > 10000 nM T02446 C2MD1Q 155513187 IC50 > 10000 nM T02446 D05FXD 44478401 IC50 = 1.1 nM T02446 D0X8BU 71718651 IC50 = 3800 nM T51565 D0K8KX 5280343 Ki = 1180 nM T51565 D09JEJ 24748573 Ki = 0.38 nM T51565 D0A5MC 11712649 IC50 = 20500 nM T51565 D0B9BU 6918454 IC50 = 17 nM T51565 D0E3TC 44259 IC50 = 3617 nM T51565 D0X5GF 9981969 Ki = 70 nM T51565 D00PWQ 3820 IC50 = 20000 nM T51565 D02GEJ 5326976 Ki = 40 nM T51565 D01LQC 24779676 Ki = 5 nM T51565 D0J0EL 2950 Ki > 40000 nM T51565 D0T3ME 156422 IC50 > 30000 nM T51565 D0U7OU 3220 IC50 = 890 nM T51565 C12LHD 5004 Ki = 60 nM T51565 C7L0IN 75358 Ki = 400 nM T51565 CFR08Z 85466 Ki = 350 nM T51565 C63WLY 89644 IC50 > 10 ug.mL-1 T51565 C5JE2Z 104860 IC50 > 10 ug.mL-1 T51565 CI1NA5 159926 IC50 > 10 ug.mL-1 T51565 CYBA43 177458 IC50 > 10 ug.mL-1 T51565 CJH12X 537952 IC50 = 26800 nM T51565 C9R7ZX 704429 IC50 = 14000 nM T51565 CDA3U5 705545 IC50 = 7000 nM T51565 C2QZL7 768039 IC50 = 6000 nM T51565 CW04CM 779228 IC50 = 27700 nM T51565 C58XVH 779231 Ki = 1600 nM T51565 CVUO95 837195 IC50 > 25000 nM T51565 CYO8Z5 877536 Ki = 1100 nM T51565 C5AJ3P 1075904 IC50 = 8000 nM T51565 CSM1Z5 3246023 IC50 = 400 nM T51565 CCZ7D1 4634231 Ki = 780 nM T51565 CTR3O2 5326637 Ki = 780 nM T51565 CDQ3M7 5359485 IC50 = 2 ug.mL-1 T51565 C54BYP 5360741 IC50 > 10 ug.mL-1 T51565 CU91NS 5382529 Ki > 40000 nM T51565 C1VZ5E 5795340 Ki = 60 nM T51565 CL01KA 7328979 IC50 = 2000 nM T51565 C2OAV0 7328982 Ki = 180 nM T51565 CL8FY5 7719528 IC50 > 50000 nM T51565 CQYD70 8244321 IC50 = 10900 nM T51565 C5YH2A 8415300 IC50 = 13000 nM T51565 C7QFS4 10423877 IC50 > 200000 nM T51565 CR9EJ0 11352337 Ki = 154 nM T51565 C8V7ZF 11352967 Ki = 106 nM T51565 CXBU49 11502255 IC50 > 100000 nM T51565 CO9KP5 11583459 IC50 > 10000 nM T51565 CCG79O 13814386 IC50 = 63 nM T51565 CDGF78 15282555 IC50 = 4100 nM T51565 CE03FU 16224058 IC50 = 2700 nM T51565 CV78IN 16224258 IC50 = 110 nM T51565 CFO0B6 16386786 IC50 = 15200 nM T51565 C2J5QI 19689569 IC50 = 3200 nM T51565 CCKJ89 19967010 IC50 = 3600 nM T51565 CP89VG 21948240 IC50 = 9600 nM T51565 COC1L6 23656870 Ki = 0.35 nM T51565 C7YG1N 24759534 IC50 = 8300 nM T51565 CML7B3 24779675 Ki = 8 nM T51565 CBP53T 24779677 Ki = 24 nM T51565 CU6V1E 24779678 Ki = 137 nM T51565 CY8X0J 24811794 IC50 = 663 nM T51565 C32SUJ 24894993 IC50 = 93000 nM T51565 CN13JF 24899915 IC50 = 2 ug.mL-1 T51565 CBWR97 24899916 IC50 > 10 ug.mL-1 T51565 C9F2JD 24899917 IC50 > 10 ug.mL-1 T51565 C64MTI 24900160 IC50 > 10 ug.mL-1 T51565 CO2I6Q 24900161 IC50 > 10 ug.mL-1 T51565 CLWA97 38326233 IC50 = 102600 nM T51565 CFS0V9 40064287 IC50 > 200000 nM T51565 C5KB4C 41470891 IC50 = 520 nM T51565 C2TJZ0 41544951 IC50 = 16100 nM T51565 CJ5U1X 42639664 IC50 > 10 ug.mL-1 T51565 CQVZ16 44123806 IC50 = 540 nM T51565 C1O6NR 44123807 IC50 = 320 nM T51565 C91MBN 44123808 IC50 = 340 nM T51565 C4HY6I 44263430 Ki = 43 nM T51565 CI29YJ 44263433 Ki = 300 nM T51565 C0OR9F 44263437 Ki = 200 nM T51565 CYX19V 44263445 Ki = 80 nM T51565 C0RK5W 44263447 Ki = 261 nM T51565 CNZ19H 44263451 Ki = 670 nM T51565 CLPT75 44426741 Ki = 168 nM T51565 CMIV60 44426742 Ki = 5 nM T51565 CZF83Q 44426743 Ki = 9 nM T51565 CG0Q6R 44426744 Ki = 23 nM T51565 C8LTP3 44426745 Ki = 45 nM T51565 C8HBL9 44426746 Ki = 55 nM T51565 CXE41T 44426747 Ki = 13 nM T51565 CIZB06 44426748 Ki = 12 nM T51565 C91PVD 44426749 Ki = 14 nM T51565 C3ZG5A 44426750 Ki = 126 nM T51565 CBS8Y1 44426751 Ki = 11 nM T51565 CIJ05K 44426752 Ki = 7 nM T51565 CRX64G 44426756 Ki = 137 nM T51565 C0WN7G 44426757 Ki = 3400 nM T51565 C61RVT 44426758 Ki = 8 nM T51565 CF3J1B 44426760 Ki = 0.26 nM T51565 CJI2F4 44426761 Ki = 1.9 nM T51565 C6LYM7 44426763 Ki = 35 nM T51565 C8JUD9 44426764 Ki = 11 nM T51565 CV7QG2 44426765 Ki = 2000 nM T51565 CE30HU 44426767 Ki = 17 nM T51565 C20UGL 44426768 Ki = 210 nM T51565 CR1U8A 44426769 Ki = 550 nM T51565 C62ICV 44426770 Ki = 500 nM T51565 CL4WS8 44426771 Ki = 95 nM T51565 CRQC42 44426773 Ki = 190 nM T51565 CP59GR 44426774 Ki = 700 nM T51565 CC18PQ 44426776 Ki = 370 nM T51565 CL3VK2 44426778 Ki = 190 nM T51565 C56ERL 44426779 Ki = 190 nM T51565 CA4JX9 44426786 Ki = 15 nM T51565 C3VRO9 44557921 IC50 > 10000 nM T51565 CF90OX 44576212 IC50 > 100000 nM T51565 CX08MT 44590715 IC50 = 9250 nM T51565 CVK4W9 44590746 IC50 = 2200 nM T51565 C3QRL8 44590749 IC50 = 11200 nM T51565 C4MY0L 44590794 IC50 = 7300 nM T51565 CLPU05 44590795 IC50 = 1730 nM T51565 C1CQS8 44590796 IC50 = 2900 nM T51565 C3F2TS 45879388 IC50 = 79300 nM T51565 CN83IB 47084137 IC50 > 200000 nM T51565 CKR3Z7 48429781 IC50 = 11500 nM T51565 CHSF07 49806372 IC50 > 1000 nM T51565 CL4FO3 50942245 IC50 = 14 nM T51565 CBC2I4 53326156 Ki = 420 nM T51565 C8NA4L 53384644 IC50 > 30000 nM T51565 CM6IZ1 54470098 Ki = 400 nM T51565 CVTQ95 56838941 Ki = 7 nM T51565 CDK93W 56946894 IC50 < 3 nM T51565 CE2DU7 56968171 Ki = 368 nM T51565 C4RIA1 56968172 Ki = 456 nM T51565 CYIO69 56968174 Ki = 116 nM T51565 CT1ZJ3 56968175 Ki = 112 nM T51565 C73NVJ 56968176 Ki = 77 nM T51565 C0MS9N 56968177 Ki = 88 nM T51565 C8WDK1 57342036 IC50 = 20 nM T51565 C0I6SZ 57342039 IC50 = 74000 nM T51565 CA7BS4 57342210 IC50 = 140 nM T51565 CVBF89 57342215 IC50 = 50000 nM T51565 C8P1ZB 57342375 IC50 = 29900 nM T51565 CH6RV3 57342376 IC50 = 4400 nM T51565 C65NOS 57342377 IC50 = 6600 nM T51565 C8TFC7 57342378 Ki = 32 nM T51565 CZ0R4K 57342379 IC50 = 6400 nM T51565 C8U4MB 57342380 IC50 = 5100 nM T51565 CJSO14 57342381 IC50 = 5100 nM T51565 CW3P9K 57342382 IC50 = 6000 nM T51565 CFX60S 57342541 IC50 = 3900 nM T51565 CF9BZ1 57342542 IC50 = 3600 nM T51565 C2C4XB 57342543 IC50 = 6800 nM T51565 C9XPF2 57342544 IC50 = 8100 nM T51565 C9MA4U 57342545 IC50 = 5700 nM T51565 CWZY51 57342546 IC50 = 14100 nM T51565 CK9IC1 57342547 IC50 = 7700 nM T51565 CO14NX 57342548 IC50 = 5100 nM T51565 CTNX36 57342718 IC50 = 4500 nM T51565 C8G6RK 57342719 IC50 = 6100 nM T51565 C8X5JG 57384039 IC50 = 10 nM T51565 CV0GJ4 57384040 IC50 = 4 nM T51565 CJ9OF3 57400663 Ki = 13 nM T51565 CXJ63M 59603829 IC50 > 100000 nM T51565 CQEU96 59603842 IC50 > 10000 nM T51565 C2JS8M 60650870 IC50 > 50000 nM T51565 CV63UL 67240318 IC50 > 10000 nM T51565 C5DGR9 69036886 IC50 = 10000 nM T51565 CR34AU 70682211 IC50 = 240 nM T51565 C4TM6F 70682212 IC50 = 10 nM T51565 C3ITR6 70682213 IC50 < 3000 nM T51565 C9PE4T 70682214 IC50 < 3 nM T51565 CW4C1K 70684312 IC50 < 3 nM T51565 C97TBH 70684313 IC50 = 24 nM T51565 CTWO98 70684314 IC50 = 83 nM T51565 CI8E0T 70686471 IC50 = 58 nM T51565 C04EAX 70686472 IC50 = 430 nM T51565 C7OX5Z 70686473 IC50 = 26 nM T51565 C34SEQ 70686474 IC50 = 860 nM T51565 CW9M8Z 70688568 IC50 = 78 nM T51565 CPQN62 70688569 IC50 = 79 nM T51565 CPT42B 70688570 IC50 = 6000 nM T51565 C9GLA0 70690634 IC50 = 100 nM T51565 CF2KQ7 70690635 IC50 = 250 nM T51565 CT5U7D 70690636 IC50 = 4 nM T51565 C3C1SY 70690637 IC50 = 500 nM T51565 C6AL5J 70690638 IC50 = 15000 nM T51565 C49HXT 70692773 IC50 = 460 nM T51565 CH7JP3 70692774 IC50 = 270 nM T51565 CXU1Q3 70692775 IC50 = 120 nM T51565 CRG53C 70694812 IC50 = 180 nM T51565 CVW72S 70694813 IC50 = 52 nM T51565 CHN90R 70696862 IC50 = 30 nM T51565 C1JH4X 70696863 IC50 = 30 nM T51565 C18WOS 70696864 IC50 = 40 nM T51565 CP08FT 70696865 IC50 = 30 nM T51565 CNM85T 71664579 IC50 = 100 nM T51565 C8S3ON 72163808 IC50 < 3 nM T51565 CPA03W 72163810 IC50 < 3 nM T51565 CR4B7C 72163925 IC50 < 3 nM T51565 CQFI71 72163926 IC50 < 3 nM T51565 CDN67F 72163927 IC50 < 3 nM T51565 CU64GF 72163928 IC50 < 3 nM T51565 CYNV72 72163929 IC50 < 3 nM T51565 CK0TQ3 72163930 IC50 < 3 nM T51565 CCHA62 72164043 IC50 < 3 nM T51565 CL8ZG2 72164044 IC50 < 3 nM T51565 CKT8P6 72164045 IC50 < 3 nM T51565 CYN73V 72164046 IC50 < 3 nM T51565 CECL46 72164047 IC50 < 3 nM T51565 CL64PN 72164048 IC50 < 3 nM T51565 CWS4E0 72164167 IC50 < 3 nM T51565 CX5OC1 72164168 IC50 < 3 nM T51565 CR2L3Z 72164169 IC50 < 3 nM T51565 CMI5D0 72164170 IC50 < 3 nM T51565 CL4PT9 72164171 IC50 < 3 nM T51565 CU76HL 72164286 IC50 < 3 nM T51565 CG4M7N 72164287 IC50 < 3 nM T51565 CZ7YO2 72164288 IC50 < 3 nM T51565 CDKV52 72164289 IC50 < 3 nM T51565 CJP4N6 72164290 IC50 < 3 nM T51565 CC8VU2 73353618 IC50 = 6 nM T51565 CDE3Y9 76321032 IC50 < 3 nM T51565 CC4F0A 78319160 IC50 > 50000 nM T51565 CO4IE9 78319161 IC50 > 50000 nM T51565 CY6LN4 78319162 IC50 > 50000 nM T51565 CH5K9E 84255281 IC50 = 3000 nM T51565 C4RTX7 84255286 IC50 = 12000 nM T51565 C2R5CD 85469599 IC50 = 800 nM T51565 CFMJ07 85469603 Ki = 1110 nM T51565 CN7HU3 86288843 IC50 > 50000 nM T51565 C5Y1WO 86288855 IC50 > 25000 nM T51565 C1HW4B 89735655 IC50 > 100000 nM T51565 CW0L1D 90654798 IC50 > 25000 nM T51565 CDF2A1 90654799 IC50 > 50000 nM T51565 CO2CU1 90654800 IC50 > 50000 nM T51565 C4NXO7 90654801 IC50 > 50000 nM T51565 CE54MK 90654802 IC50 > 50000 nM T51565 C5PO6N 90654803 IC50 > 25000 nM T51565 CID9U2 90654804 IC50 > 50000 nM T51565 CDU21W 118710263 IC50 = 5400 nM T51565 CS39QV 118710264 IC50 = 5600 nM T51565 C6E8JQ 118710265 IC50 = 7350 nM T51565 C2WCN1 118710266 IC50 = 4160 nM T51565 CFD05M 118710267 IC50 = 2500 nM T51565 CK87BW 118710268 IC50 = 2500 nM T51565 COI2N4 118710269 IC50 = 3600 nM T51565 CXC9M8 118710271 IC50 = 2170 nM T51565 C3KLI5 118723185 IC50 > 100000 nM T51565 CSE0M8 121232389 IC50 = 370 nM T51565 C0Q9RL 121551752 IC50 > 200000 nM T51565 C4T7YB 127025199 IC50 = 17 nM T51565 CP02TW 127025200 IC50 = 14 nM T51565 C57ECS 127025201 IC50 = 1300 nM T51565 CP31UE 127025202 IC50 = 15 nM T51565 CHP6R9 127025499 IC50 = 19 nM T51565 CY37QE 127025500 IC50 = 28 nM T51565 CR59LY 127026094 IC50 = 15 nM T51565 CWIG59 127026095 IC50 = 16 nM T51565 C45BZG 127026096 IC50 = 330 nM T51565 C0HLT9 127026097 IC50 = 26 nM T51565 CW5JB1 127026098 IC50 = 17 nM T51565 C1A4IY 127026345 Ki = 1270 nM T51565 C1OI6B 127026659 Ki = 2770 nM T51565 CS95XR 127026660 Ki = 2490 nM T51565 CJ04NV 127026661 Ki = 5030 nM T51565 CL52EB 127026662 Ki = 2420 nM T51565 CL4CG5 127026727 IC50 = 14 nM T51565 CO6X5B 127026728 IC50 = 16 nM T51565 CA5XG8 127026729 IC50 = 15 nM T51565 C6EIR3 127027657 IC50 = 14 nM T51565 C1MF5T 127029513 IC50 = 14 nM T51565 C6OTW1 127031797 Ki = 150 nM T51565 CS3Z5P 127037009 Ki = 1630 nM T51565 CZD87E 127037084 IC50 < 10000 nM T51565 C9CYG7 127037156 Ki = 2510 nM T51565 CVH94O 127037627 Ki = 1420 nM T51565 CB9Z0V 127038973 IC50 < 10000 nM T51565 C5R6YK 127043054 IC50 < 3 nM T51565 C84LJK 127043055 IC50 = 5 nM T51565 C41JXY 127043056 IC50 < 3 nM T51565 CY6Z7G 127043251 IC50 < 3 nM T51565 CF8BI9 127045382 IC50 = 9 nM T51565 CI74KJ 127045531 IC50 = 41 nM T51565 CJW82G 127045532 IC50 = 9 nM T51565 C6JB0N 127045533 IC50 < 3 nM T51565 C9YZE3 127045534 IC50 = 13 nM T51565 CRZV34 127045535 IC50 < 3 nM T51565 C6FV8P 127045536 IC50 = 6 nM T51565 C5M6AQ 127045537 IC50 < 3 nM T51565 C5SUZ1 127045538 IC50 = 6 nM T51565 C0WB6T 127045542 IC50 = 4 nM T51565 C2FW3P 127045543 IC50 < 3 nM T51565 C7WS3U 127045544 IC50 < 3 nM T51565 CGL80Q 127053115 IC50 = 16900 nM T51565 CKB5T4 127053116 IC50 = 20000 nM T51565 CDZX63 132281899 IC50 = 7000 nM T51565 C4Q5LF 132471857 IC50 = 5 nM T51565 C2AN7T 134611886 IC50 > 100000 nM T51565 CW0P1Q 135433657 IC50 > 10000 nM T51565 CZ7EX0 136183413 IC50 > 30000 nM T51565 CY36QB 136254272 IC50 = 5000 nM T51565 CPI1U0 137631770 IC50 = 300 nM T51565 C23HSQ 137651463 IC50 = 4 nM T51565 C38PAN 139593286 IC50 > 50000 nM T51565 CPL8X0 139593287 Ki = 700 nM T51565 CV28AL 145967603 IC50 = 460 nM T51565 C5B0QL 145967935 IC50 = 15 nM T51565 CMG01Q 145968043 IC50 = 130 nM T51565 C9LBY8 145968158 IC50 = 4800 nM T51565 C6RZN1 145968179 IC50 = 4600 nM T51565 CPET15 145968269 IC50 = 360 nM T51565 C24AQX 145968504 IC50 = 2700 nM T51565 CTY0I5 145968604 IC50 = 112 nM T51565 CL07SI 145968637 IC50 = 5 nM T51565 C7B3UD 145968656 IC50 = 1000 nM T51565 CZN38I 145969224 IC50 = 13000 nM T51565 CL8V5N 145969695 IC50 = 13000 nM T51565 CAU16Y 145969796 IC50 = 26 nM T51565 CISA20 145969798 IC50 > 30000 nM T51565 CZ8NL7 145969872 IC50 = 70 nM T51565 CM6D9P 145969896 IC50 > 30000 nM T51565 CT3N9K 145970124 IC50 = 20000 nM T51565 CQR9Z4 145970125 IC50 = 3 nM T51565 CPX3N9 145970645 IC50 = 360 nM T51565 CP0M6D 145970925 IC50 = 310 nM T51565 CQ4WO3 145971039 IC50 = 7 nM T51565 CD97BO 145971046 IC50 > 30000 nM T51565 C09DLU 145971051 IC50 = 297 nM T51565 CIR5M6 145980012 IC50 = 1900 nM T51565 CT02VJ 145981438 IC50 = 4000 nM T51565 CU1RE3 145981895 IC50 = 12400 nM T51565 CK5M9W 145987607 IC50 = 20400 nM T51565 CM9F8Z 145987956 IC50 = 560 nM T51565 CD7K3H 145988440 IC50 = 4600 nM T51565 C4P8SD 145989719 IC50 > 30000 nM T51565 CN6C4X 145990029 IC50 = 7900 nM T51565 CW5H3N 145990758 IC50 = 2800 nM T51565 CLF28N 145992533 IC50 = 4900 nM T51565 C2MD1Q 155513187 IC50 > 10000 nM T51565 C1PKJ8 155515774 IC50 = 5000 nM T51565 C2D1US 155516813 Ki = 220 nM T51565 C86HPW 155518524 IC50 > 100000 nM T51565 CPW3B7 155528606 IC50 > 50000 nM T51565 C1Q2ZA 155533799 IC50 > 25000 nM T51565 C8MD9V 155538565 IC50 = 5000 nM T51565 CTZ8C0 155546940 IC50 = 8000 nM T51565 C2OBT0 155550745 IC50 = 14000 nM T51565 CYZ62M 155556465 IC50 = 4000 nM T51565 COQ52X 155557908 IC50 = 8000 nM T51565 D00ERW 44444843 Ki > 5833 nM T51565 D00RIX 5280443 Ki = 740 nM T51565 D02DML 5281707 Ki = 7670 nM T51565 D02XHC 448912 IC50 >= 100000 nM T51565 D04BNM 5894 Ki = 4500 nM T51565 D04TPA 72163809 IC50 < 3 nM T51565 D06KDU 16760346 Ki = 77 nM T51565 D06QWO 14824655 IC50 > 10 ug.mL-1 T51565 D09ZNV 447682 Ki = 170 nM T51565 D0A1CM 5281855 Ki = 20 nM T51565 D0CP3M 5149739 Ki = 40 nM T51565 D0F0AX 135413546 IC50 = 7000 nM T51565 D0G3SZ 6918469 IC50 > 10 ug.mL-1 T51565 D0K6BI 46943415 Ki = 83 nM T51565 D0MF5Y 5281614 Ki = 350 nM T51565 D0O1YH 1694 Ki = 300 nM T51565 D0US9O 45275255 IC50 > 30000 nM T51565 D0Z5TQ 5924208 IC50 = 279 nM T68470 D00KHM 16362 IC50 = 2000 nM T68470 CE2DF1 509070 IC50 = 544 nM T68470 CSI70A 2307331 IC50 = 888 nM T68470 D00TFA 3392731 IC50 = 5000 nM T68470 D0M5FO 60167849 IC50 > 200000 nM T93716 D0V2YJ 11655511 IC50 > 50000 nM T93716 CTE52X 22577556 IC50 = 50000 nM T93716 CPLY38 25164463 IC50 > 50000 nM T93716 CAXQ03 25164661 IC50 > 50000 nM T93716 CRU76E 25164662 IC50 > 50000 nM T93716 C3NVW5 25165471 IC50 > 50000 nM T93716 CV6Y1Z 25165472 IC50 > 50000 nM T93716 CVMZ57 25165473 IC50 > 50000 nM T93716 CF9KY4 25165474 IC50 > 50000 nM T93716 CIWL28 25165475 IC50 > 50000 nM T93716 CPV3O6 25165666 IC50 > 50000 nM T93716 C56QHJ 25165854 IC50 > 50000 nM T93716 C1FCO0 45266928 IC50 > 50000 nM T93716 C1Y4KO 45267020 IC50 > 50000 nM T93716 CLK10E 45267851 IC50 > 50000 nM T93716 C53DIE 45267853 IC50 > 50000 nM T93716 CO5BT3 45267860 IC50 > 50000 nM T93716 C93RCK 45267863 IC50 > 50000 nM T93716 CK60GY 45267896 IC50 > 50000 nM T93716 C71NGE 45268737 IC50 > 50000 nM T93716 C2ZN5S 45268741 IC50 > 50000 nM T93716 CP4M3X 45268781 IC50 > 50000 nM T93716 C9GJA6 45269595 IC50 > 50000 nM T93716 CTW13H 45269596 IC50 > 50000 nM T93716 C96UFG 45270431 IC50 > 50000 nM T93716 CZ5ID2 45271261 IC50 > 50000 nM T93716 C0X5FN 45271263 IC50 > 50000 nM T93716 CER7W9 45271267 IC50 > 50000 nM T93716 C32JIV 45271285 IC50 > 50000 nM T93716 CN32MP 45272152 IC50 > 50000 nM T93716 CATM09 45272155 IC50 > 50000 nM T93716 C70MZU 45272180 IC50 > 50000 nM T93716 C3SRC5 45272183 IC50 > 50000 nM T93716 CRT26A 45272991 IC50 > 50000 nM T93716 CG9XA3 45272994 IC50 > 50000 nM T80975 D01PZD 5329098 IC50 = 12.9 nM T80975 D01ZRI 6450551 IC50 = 0.2 nM T80975 D03MNN 11341869 IC50 > 1000 nM T80975 D03ZBT 11626560 IC50 > 10000 nM T80975 D04LVK 57379345 IC50 = 4210 nM T80975 D07NVU 9829523 IC50 = 250 nM T80975 D07POC 176870 IC50 = 50.12 nM T80975 D08CDI 208908 IC50 > 10000 nM T80975 D09GDD 11167602 IC50 = 4.2 nM T80975 D09XZB 123631 IC50 = 48.5 nM T80975 D0AZ3C 5291 IC50 > 25000 nM T80975 D0E6XR 3062316 IC50 = 2360 nM T80975 D0E7PQ 5311 IC50 > 10000 nM T80975 D0G6QF 3081361 IC50 = 9 nM T80975 D0H0EQ 24826799 IC50 = 1.5 nM T80975 D0IQ6P 25102847 IC50 = 0.035 nM T80975 D0J1MI 4030 IC50 = 3600 nM T80975 D0J9ZR 4477 IC50 = 23100 nM T80975 D0K8KX 5280343 IC50 = 280 nM T80975 D0R0FO 9823820 IC50 = 0.7 nM T80975 D0R0MW 5329102 Ki = 2.9 nM T80975 D0SZ6E 45139106 IC50 = 1 nM T80975 D0U3SY 49806720 IC50 = 1400 nM T80975 D0W5HK 216239 Ki = 0.021 nM T80975 D0Y9EW 42611257 IC50 = 360 nM T80975 D00DRL 44137946 IC50 = 44 nM T80975 D00YPR 9811611 IC50 = 11 nM T80975 D02NNV 3038525 IC50 > 5000 nM T80975 D02RJY 11442891 IC50 = 432 nM T80975 D02UFQ 11620908 IC50 > 10000 nM T80975 D02WVT 25031915 IC50 = 25 nM T80975 D03AND 11656518 IC50 = 1300 nM T80975 D03HUX 49792852 IC50 > 10000 nM T80975 D03LWG 53235510 IC50 = 180 nM T80975 D03QLG 9917013 IC50 = 43 nM T80975 D04AHQ 71721540 IC50 = 3900 nM T80975 D04OTY 24756034 IC50 = 1.3 nM T80975 D05PCM 78323835 IC50 = 1200 nM T80975 D05PZB 135398495 IC50 = 10 nM T80975 D06KTJ 53252276 IC50 = 88 nM T80975 D06TFI 10090485 IC50 = 442 nM T80975 D07EHV 44814409 IC50 > 10000 nM T80975 D07HPJ 11476171 IC50 = 7100 nM T80975 D07HRU 9549295 IC50 = 1 nM T80975 D07KYT 24889392 IC50 = 430 nM T80975 D07NOI 9808844 IC50 = 6 nM T80975 D07NUL 118414016 IC50 = 5330 nM T80975 D07PNT 10433653 IC50 = 6 nM T80975 D08FDX 24901704 IC50 = 6 nM T80975 D08HOM 46207586 IC50 = 3 nM T80975 D09ETH 16118392 IC50 = 16 nM T80975 D09VMI 9933475 IC50 = 0.5 nM T80975 D0A1AQ 5329099 IC50 = 2430 nM T80975 D0AX4H 78427026 IC50 = 109 nM T80975 D0CY1B 6420138 Ki = 44 nM T80975 D0D1GF 42642645 IC50 = 0.8 nM T80975 D0D4VV 46944259 IC50 = 5.8 nM T80975 D0E3TC 44259 IC50 = 1.2 nM T80975 D0E5XA 11569967 IC50 = 19 nM T80975 D0FA6S 54576299 IC50 = 9.2 nM T80975 D0FD6D 11751922 IC50 = 4 nM T80975 D0G2QH 10297043 IC50 = 77 nM T80975 D0G9AW 59473233 EC50 > 1000 nM T80975 D0GP9Q 11973736 IC50 >= 10000 nM T80975 D0H2HZ 60194098 IC50 = 31622.78 nM T80975 D0H9FR 118295624 IC50 = 705 nM T80975 D0HS5V 11234052 Ki = 26 nM T80975 D0M0XB 10302451 IC50 = 20900 nM T80975 D0M9QZ 11485656 IC50 = 2.3 nM T80975 D0MR0B 54766013 IC50 = 97 nM T80975 D0N8RV 9868037 IC50 = 9 nM T80975 D0NW0T 67462786 IC50 = 36.8 nM T80975 D0O0LS 25141092 IC50 > 1000 nM T80975 D0O6WV 24794418 IC50 = 138.7 nM T80975 D0P1CV 46191454 IC50 > 10000 nM T80975 D0P6DJ 151194 IC50 < 15 nM T80975 D0Q7RE 16007391 Ki = 1800 nM T80975 D0Q9CY 9915743 IC50 = 858.2 nM T80975 D0Q9UX 16718576 IC50 > 10000 nM T80975 D0S3PO 6445562 IC50 = 3131 nM T80975 D0S6TK 11213558 EC50 = 36 nM T80975 D0S7HM 16041424 IC50 = 10 nM T80975 D0T2ER 24767976 IC50 = 0.95 nM T80975 D0VF6E 1401 EC50 = 250 nM T80975 D0W7JZ 9911830 IC50 = 0.16 nM T80975 D0XT0W 66555680 IC50 = 2100 nM T80975 D0Z1DH 10029385 IC50 > 20000 nM T80975 D0Z4RC 24756910 IC50 = 849 nM T80975 D0Z6MT 16662431 IC50 = 5 nM T80975 D0ZN1R 68245 IC50 = 5.09 nM T80975 D03BNU 59604787 IC50 > 3500 nM T80975 D0LF0O 135441202 IC50 = 369 nM T80975 D00PWQ 3820 IC50 > 100000 nM T80975 D04SWX 56924694 IC50 = 34 nM T80975 D0JY1I 42613483 IC50 = 11000 nM T80975 D0YK9D 9956119 IC50 > 5000 nM T80975 D00DQX 11667893 IC50 = 3 nM T80975 D04FHB 6918852 Ki > 5000 nM T80975 D06GBK 2048 IC50 = 6200 nM T80975 D09HEV 6539952 IC50 = 1190 nM T80975 D0H4GI 10275001 IC50 = 8 nM T80975 D0IT6Q 3038522 IC50 = 2070 nM T80975 D0L5YF 5329032 IC50 = 30 nM T80975 D0Q7HO 4705 IC50 = 1489 nM T80975 D0T3ME 156422 IC50 = 340 nM T80975 CB1VW3 1400 IC50 = 1600 nM T80975 C8HN2C 3798 IC50 = 7000 nM T80975 C63WLY 89644 IC50 = 7.3 ug.mL-1 T80975 CE4K5D 92516 IC50 > 50000 nM T80975 C5JE2Z 104860 IC50 = 1.4 ug.mL-1 T80975 C6Y9CV 151193 IC50 = 37 nM T80975 CI1NA5 159926 IC50 = 2.4 ug.mL-1 T80975 CI80NA 160436 IC50 > 50000 nM T80975 CYBA43 177458 IC50 = 1.2 ug.mL-1 T80975 CHR70B 237859 IC50 = 140000 nM T80975 CO6B3I 265711 IC50 = 21600 nM T80975 CV3XI1 354479 IC50 = 200 nM T80975 CKJ1B7 382514 IC50 = 66000 nM T80975 CN05AH 406563 IC50 = 8.5 nM T80975 CK0L4O 442514 IC50 = 2100 nM T80975 C9E4FI 447622 IC50 = 148 nM T80975 C1ZG2U 449087 IC50 > 10000 nM T80975 C18WEB 490561 IC50 = 43 nM T80975 C5NRQ2 619921 IC50 = 124 nM T80975 CEG3W5 657169 IC50 = 16.5 nM T80975 C6CJY8 725409 IC50 > 10000 nM T80975 CK5OB3 769922 IC50 = 112.7 nM T80975 CW75ZS 787612 IC50 > 10000 nM T80975 CXK7Y3 787613 IC50 > 10000 nM T80975 C7L1YW 792771 IC50 = 23.6 nM T80975 CSQ76E 836104 IC50 = 134.6 nM T80975 C46VKZ 836113 IC50 = 124.6 nM T80975 CCT7R0 837055 IC50 = 208.8 nM T80975 CDSN72 838889 IC50 = 1122.02 nM T80975 CW7S5J 980157 IC50 = 5.9 nM T80975 C5C3ZL 1036473 IC50 = 4.1 nM T80975 C2DI6O 1107690 IC50 = 2.9 nM T80975 C9VF7N 1109437 IC50 = 400 nM T80975 CHK0M3 1132697 IC50 = 5 nM T80975 C5SUY7 1146874 IC50 > 10000 nM T80975 CHW5G2 1386118 IC50 = 1700 nM T80975 CB2V1M 1386625 IC50 > 10000 nM T80975 CA67ZG 1391316 IC50 = 2000 nM T80975 C9C8DI 1393513 IC50 = 840 nM T80975 CNF37I 1419346 IC50 > 10000 nM T80975 CT1M4K 1419523 IC50 = 6900 nM T80975 CGA05N 1462274 IC50 = 10 nM T80975 COB86I 1474850 IC50 = 2900 nM T80975 CJP04L 1474852 IC50 = 800 nM T80975 CIPW30 1474854 IC50 = 2900 nM T80975 C2GSN6 1475052 IC50 = 800 nM T80975 CBU82E 1918383 IC50 > 10000 nM T80975 CJO12B 2132378 IC50 = 5.6 nM T80975 C1SVD2 2132479 IC50 = 1300 nM T80975 CAV19R 2360773 IC50 > 10000 nM T80975 C6T0OJ 2400783 IC50 > 10000 nM T80975 C4MZU7 2803617 IC50 > 50000 nM T80975 C8S0UP 2806990 IC50 = 7730 nM T80975 C2AFE3 2808988 IC50 = 4800 nM T80975 C9Z1FJ 2810885 IC50 = 92700 nM T80975 CH4V8I 2811823 IC50 = 51600 nM T80975 CH64KM 2814387 IC50 = 47000 nM T80975 CI6VH2 2817227 IC50 = 17800 nM T80975 CLM4F6 2869439 IC50 > 10000 nM T80975 CAT3C7 2885152 IC50 > 10000 nM T80975 C3BJP7 2943601 IC50 = 3500 nM T80975 CHC5I0 2971839 IC50 > 10000 nM T80975 CFY1D0 2974957 IC50 > 10000 nM T80975 CFVK40 3008950 IC50 = 5080 nM T80975 CD8UW1 3008956 IC50 = 28100 nM T80975 CCD93P 3008957 IC50 > 50000 nM T80975 CU64VM 3008958 IC50 > 50000 nM T80975 C8F0KM 3008959 IC50 = 5580 nM T80975 CV8R9Z 3008960 IC50 = 5970 nM T80975 C8EZ6O 3008961 IC50 = 250 nM T80975 CX95SU 3008962 IC50 = 620 nM T80975 C9B2MN 3008963 IC50 = 8280 nM T80975 C9E7BW 3008964 IC50 > 50000 nM T80975 CGK91Q 3008965 IC50 = 9420 nM T80975 CCN9D5 3142817 IC50 = 3000 nM T80975 CQ3YR1 3262021 IC50 > 10000 nM T80975 CG0KP8 3472544 IC50 = 4900 nM T80975 C4P8KQ 3889479 IC50 = 1100 nM T80975 CS64FZ 4118382 IC50 = 930 nM T80975 CP3C4Y 4165705 IC50 = 100000 nM T80975 CUV81H 4182686 IC50 = 4700 nM T80975 CPN2S0 4369497 IC50 = 17.1 nM T80975 CI4C6L 4561389 IC50 = 1274 nM T80975 C8O9MN 4616059 IC50 > 10000 nM T80975 CW7IX9 4647210 IC50 = 88.5 nM T80975 CB3G6R 4913175 IC50 = 30 nM T80975 CDE83C 5136768 IC50 = 107.2 nM T80975 CH1G9Q 5147149 IC50 = 54 nM T80975 C8T6DH 5147155 IC50 = 830 nM T80975 CJDO18 5147157 IC50 = 110 nM T80975 C8IAR2 5281657 IC50 = 11700 nM T80975 CI68PW 5283685 IC50 = 6010 nM T80975 CXK0S6 5283727 IC50 = 4350 nM T80975 CFPX04 5292020 IC50 > 10000 nM T80975 C5BMS3 5292021 IC50 > 10000 nM T80975 COS56T 5292024 IC50 > 10000 nM T80975 C86DQC 5292025 IC50 > 10000 nM T80975 CJ9R3P 5292026 IC50 > 10000 nM T80975 CV2M9N 5292027 IC50 > 10000 nM T80975 CYBL90 5292028 IC50 > 10000 nM T80975 CVT10F 5292029 IC50 = 630 nM T80975 CNZ3D6 5298697 IC50 = 470 nM T80975 CT40IY 5298699 IC50 > 10000 nM T80975 CMFK67 5298701 IC50 > 10000 nM T80975 CA0LO9 5298702 IC50 > 10000 nM T80975 C0RXL8 5326956 IC50 = 3 nM T80975 CKY7Z5 5328227 IC50 > 10000 nM T80975 CWX63A 5329004 IC50 = 9 nM T80975 CQL3C9 5329005 IC50 = 2700 nM T80975 CFW19M 5329009 IC50 = 510 nM T80975 C2FO4B 5329010 IC50 = 2.3 nM T80975 CZU0K3 5329011 IC50 = 7 nM T80975 C21WXV 5329012 IC50 < 5 nM T80975 CJ68OQ 5329013 IC50 < 2 nM T80975 CEJR83 5329014 IC50 = 60 nM T80975 COS5M9 5329015 IC50 = 150 nM T80975 CKFS07 5329016 IC50 < 2 nM T80975 CC1EO4 5329017 IC50 = 10 nM T80975 CGC01T 5329018 IC50 = 40 nM T80975 C1XJL0 5329019 IC50 = 40 nM T80975 C9SZ4Q 5329020 IC50 = 9 nM T80975 C5DO1Y 5329021 IC50 = 40 nM T80975 C2YDI8 5329022 IC50 = 60 nM T80975 CW3OV5 5329023 IC50 = 8 nM T80975 C6HSX8 5329024 IC50 = 60 nM T80975 CP37NS 5329025 IC50 = 40 nM T80975 C3VHF6 5329026 IC50 = 6 nM T80975 CSRF48 5329027 IC50 = 100 nM T80975 CB6V5Y 5329028 IC50 = 10 nM T80975 C6AN1O 5329029 IC50 > 100000 nM T80975 C04EAP 5329030 IC50 = 1500 nM T80975 C1Y5QP 5329031 IC50 = 300 nM T80975 C4VLR8 5329033 IC50 = 40 nM T80975 CLT7J9 5329034 IC50 = 300 nM T80975 C9VX8C 5329040 IC50 = 230 nM T80975 CK6T4U 5329042 IC50 = 25 nM T80975 CA81XO 5329045 IC50 = 25 nM T80975 C4T3MO 5329046 IC50 = 10 nM T80975 CQ15KR 5329049 IC50 = 30 nM T80975 C49KNS 5329050 IC50 = 40 nM T80975 C3C1EZ 5329051 IC50 = 15 nM T80975 C0H5XL 5329052 IC50 = 55 nM T80975 CW0KA8 5329053 IC50 = 6 nM T80975 COEN93 5329054 IC50 = 40 nM T80975 CATX52 5329055 IC50 = 5 nM T80975 CEQP41 5329056 IC50 = 1 nM T80975 CDV4C9 5329057 IC50 = 10 nM T80975 C9I7WT 5329100 IC50 = 300 nM T80975 CMWB28 5329101 IC50 = 50 nM T80975 CGX50J 5329104 IC50 = 32 nM T80975 C2VX0H 5329105 IC50 = 80 nM T80975 CK71MQ 5329106 IC50 = 60 nM T80975 CL0Q4S 5329107 IC50 = 25 nM T80975 C6YRH8 5329108 IC50 = 90 nM T80975 CFP59Y 5329109 IC50 < 160 nM T80975 C0JW3Y 5329134 IC50 = 200 nM T80975 CO7J2A 5329135 IC50 = 40 nM T80975 CQ4TP5 5329136 IC50 = 28300 nM T80975 CXQC42 5329137 IC50 = 460 nM T80975 CT94JS 5329138 IC50 = 400 nM T80975 CNH06M 5329139 IC50 = 240 nM T80975 CRY4Z2 5329140 IC50 = 920 nM T80975 CAPE50 5329141 IC50 = 1350 nM T80975 CFU58A 5329142 IC50 = 300 nM T80975 C5Q8XK 5329143 IC50 = 90 nM T80975 C8PX4D 5329144 IC50 = 40 nM T80975 C6USQ5 5329145 IC50 = 1800 nM T80975 C56LWT 5329146 IC50 = 70 nM T80975 CZ16MN 5329147 IC50 = 70 nM T80975 CAN16I 5329148 IC50 = 1260 nM T80975 CG4NC2 5329149 IC50 = 670 nM T80975 CIW70H 5329150 IC50 = 140 nM T80975 C5FT6A 5329151 IC50 = 300 nM T80975 CB0N4L 5329152 IC50 = 3000 nM T80975 COFP24 5329153 IC50 = 520 nM T80975 CGWD98 5329154 IC50 = 480 nM T80975 C4PD0K 5329156 IC50 = 30 nM T80975 C0RWT8 5329157 IC50 = 20 nM T80975 C3MU5S 5329158 IC50 = 12100 nM T80975 CN6O4R 5329159 IC50 > 20000 nM T80975 CG68DI 5329160 IC50 > 20000 nM T80975 CYR7V0 5329161 IC50 = 20000 nM T80975 C9BXE2 5329162 IC50 > 20000 nM T80975 CY4V5Z 5329163 IC50 = 90 nM T80975 CI64YA 5329164 IC50 = 30 nM T80975 C2ZV0O 5329165 IC50 = 600 nM T80975 CAB53L 5329166 IC50 = 4 nM T80975 CTW9R8 5329167 IC50 = 380 nM T80975 C8A3TJ 5329168 IC50 = 50 nM T80975 CVTD82 5329169 IC50 = 70 nM T80975 CQ5WK1 5329170 IC50 = 60 nM T80975 CNC9T7 5329171 IC50 = 30 nM T80975 C6L0UW 5329229 IC50 > 20000 nM T80975 C1DBV6 5329230 IC50 > 20000 nM T80975 CLKM80 5329231 IC50 = 3470 nM T80975 CTQ18A 5329232 IC50 = 16500 nM T80975 CM5KG6 5329233 IC50 > 20000 nM T80975 CQG6R2 5329234 IC50 = 8920 nM T80975 CJ3A9I 5329235 IC50 > 20000 nM T80975 CPS7X1 5329236 IC50 > 20000 nM T80975 CAN60T 5329237 IC50 = 5820 nM T80975 CY15JP 5329238 IC50 = 10100 nM T80975 C41UBI 5329239 IC50 > 20000 nM T80975 C6VQ9F 5329240 IC50 > 20000 nM T80975 C8WS5K 5329241 IC50 > 20000 nM T80975 CI26UN 5329242 IC50 > 20000 nM T80975 C6PJ2R 5329243 IC50 > 20000 nM T80975 C0OKB7 5329244 IC50 = 300 nM T80975 C78ZNL 5329245 IC50 = 1630 nM T80975 CWL5S4 5329246 IC50 = 360 nM T80975 C4X3OE 5329248 IC50 = 40 nM T80975 CK8FH6 5329249 IC50 = 3460 nM T80975 CN5B6C 5329250 IC50 = 2050 nM T80975 CQ0B6E 5329251 IC50 = 2100 nM T80975 C4KO3N 5329252 IC50 = 3470 nM T80975 C6MZF8 5329253 IC50 > 20000 nM T80975 CBYM90 5329323 IC50 = 7 nM T80975 CXK9U6 5329324 IC50 = 6 nM T80975 CG12LJ 5329325 IC50 = 3 nM T80975 CRZ24K 5329326 IC50 = 28 nM T80975 C2S0ZV 5329327 IC50 = 2 nM T80975 CMN3H7 5329328 IC50 = 13 nM T80975 C9TD7V 5329329 IC50 = 13 nM T80975 CN7E2P 5329330 IC50 = 8 nM T80975 C8PF4Q 5329331 IC50 = 47 nM T80975 C9OB6X 5329332 IC50 = 28 nM T80975 CA7UL5 5329333 IC50 = 12 nM T80975 CL35MR 5329334 IC50 = 9 nM T80975 C70WCS 5329335 IC50 = 48 nM T80975 COQ41S 5329336 IC50 = 12 nM T80975 CKD3W6 5329337 IC50 = 71 nM T80975 C7RSX1 5329339 IC50 = 98 nM T80975 C2FT3V 5329340 IC50 = 145 nM T80975 CYF4N7 5329341 IC50 = 930 nM T80975 C54EMB 5329342 IC50 = 242 nM T80975 C30KEL 5329343 IC50 = 2840 nM T80975 CA6V9M 5329344 IC50 = 42 nM T80975 CTBN17 5329345 IC50 = 99 nM T80975 C49IYB 5329346 IC50 = 50 nM T80975 CU1Y0L 5329347 IC50 = 77 nM T80975 CPK3S2 5329348 IC50 = 52 nM T80975 CL3JM1 5329349 IC50 = 69 nM T80975 C7GRL3 5329350 IC50 = 13 nM T80975 CV98DI 5329351 IC50 = 28 nM T80975 CB72RL 5329352 IC50 = 120 nM T80975 C6QJS4 5329353 IC50 = 96 nM T80975 C81MKD 5329354 IC50 = 67 nM T80975 CS1OP7 5329355 IC50 = 186 nM T80975 CXUO96 5329356 IC50 = 575 nM T80975 CCAX78 5329357 IC50 = 5700 nM T80975 C02WSO 5329358 IC50 = 8320 nM T80975 CQU2F4 5329359 IC50 = 4860 nM T80975 CSD46A 5329360 IC50 = 4040 nM T80975 C5VIZ2 5329362 IC50 = 115 nM T80975 C51WBJ 5329363 IC50 = 111 nM T80975 CNYT34 5329364 IC50 = 60 nM T80975 C9ZPN1 5329365 IC50 = 38 nM T80975 CFDU12 5329366 IC50 = 16 nM T80975 CPMR59 5329367 IC50 = 64 nM T80975 CH19WM 5329368 IC50 = 46 nM T80975 COC9Q6 5329372 IC50 = 7 nM T80975 CJF4G6 5329373 IC50 = 4 nM T80975 CV6Z8M 5329374 IC50 = 8 nM T80975 C7H9WF 5329375 IC50 = 4 nM T80975 C6Z4BY 5329376 IC50 = 5 nM T80975 CQ9PE4 5329377 IC50 = 5 nM T80975 CC59GQ 5329378 IC50 = 5 nM T80975 CVH5Z9 5329379 IC50 = 6 nM T80975 C5ZP2J 5329380 IC50 = 10 nM T80975 C2TM0N 5329381 IC50 = 11 nM T80975 CI8YN5 5329382 IC50 = 16 nM T80975 CJY0X6 5329383 IC50 = 14 nM T80975 C2EO9W 5329384 IC50 = 151 nM T80975 C7IZ1P 5329385 IC50 = 81 nM T80975 CJXC61 5329386 IC50 = 23 nM T80975 CCX78N 5329387 IC50 = 36 nM T80975 CLN4K9 5329388 IC50 = 137 nM T80975 C1RJL7 5329389 IC50 = 240 nM T80975 CIM93H 5329390 IC50 = 259 nM T80975 C8SZO5 5329391 IC50 = 13 nM T80975 C2X3NG 5329392 IC50 = 6 nM T80975 C5TV3I 5329393 IC50 = 19 nM T80975 CRG50D 5329394 IC50 = 10 nM T80975 CIK02H 5329395 IC50 = 35 nM T80975 CK7C5S 5329396 IC50 = 14 nM T80975 CIM4F2 5329397 IC50 = 46 nM T80975 C0CAQ9 5329398 IC50 = 11 nM T80975 CYZ6V7 5329399 IC50 = 3 nM T80975 CM98VE 5329400 IC50 = 71 nM T80975 C4WZC3 5329401 IC50 = 194 nM T80975 CG0C1I 5329402 IC50 = 36 nM T80975 CT60OL 5329403 IC50 = 1880 nM T80975 CRM89A 5329405 IC50 = 23 nM T80975 CEV51Q 5329406 IC50 = 52 nM T80975 C26AUJ 5329407 IC50 = 25 nM T80975 CI2FY6 5329408 IC50 = 37 nM T80975 C6J5VL 5329409 IC50 = 88 nM T80975 CH9V0R 5329410 IC50 = 270 nM T80975 C0Z6KP 5329411 IC50 = 96 nM T80975 CK01UR 5329412 IC50 = 14 nM T80975 CGMC45 5329413 IC50 = 37 nM T80975 C7JOT5 5329414 IC50 = 3080 nM T80975 CYN3I2 5329415 IC50 = 18 nM T80975 CZIX74 5329416 IC50 = 279 nM T80975 COM81Z 5329417 IC50 = 6 nM T80975 CTWV16 5329418 IC50 = 289 nM T80975 CKF1O7 5329419 IC50 = 20 nM T80975 CSYH72 5329420 IC50 = 392 nM T80975 C7WEG5 5329421 IC50 = 5 nM T80975 CW4KM0 5329422 IC50 = 25 nM T80975 C73GBF 5329423 IC50 = 26 nM T80975 CZP9C6 5329424 IC50 = 10 nM T80975 CS9U4Q 5329425 IC50 = 77 nM T80975 C9MZ2K 5329426 IC50 = 5 nM T80975 CF6RU3 5329427 IC50 = 19000 nM T80975 CU5IV8 5329428 IC50 = 9 nM T80975 CB8O7C 5329429 IC50 = 32 nM T80975 CS0OH5 5329430 IC50 = 6830 nM T80975 C43DFA 5329431 IC50 = 340 nM T80975 CGA81W 5329432 IC50 = 273 nM T80975 C28BDN 5329433 IC50 = 3570 nM T80975 CV1S5R 5329434 IC50 = 276.5 nM T80975 C5TA0S 5329435 IC50 = 135 nM T80975 C2U3MT 5329436 IC50 = 1610 nM T80975 C0NS1F 5329437 IC50 = 2390 nM T80975 CPK05F 5329438 IC50 = 1410 nM T80975 C8C4WM 5329439 IC50 = 149 nM T80975 C8C6SL 5329440 IC50 = 45 nM T80975 CX1HJ7 5329441 IC50 = 1870 nM T80975 CMSD45 5329442 IC50 = 60 nM T80975 CZ4L3I 5329443 IC50 = 765 nM T80975 C7O9TV 5329444 IC50 = 4220 nM T80975 CS6G5X 5329445 IC50 = 232 nM T80975 CI4TV0 5329446 IC50 = 4 nM T80975 CWYP60 5329447 IC50 = 9 nM T80975 CHPC19 5329448 IC50 = 14 nM T80975 C21ZFW 5329449 IC50 = 10 nM T80975 CR4D1V 5329451 IC50 = 19 nM T80975 CKT02A 5329452 IC50 = 20 nM T80975 C4RUV5 5329453 IC50 = 11 nM T80975 CWMY68 5329455 IC50 = 113 nM T80975 CC5GB6 5329456 IC50 = 62 nM T80975 CGN7B0 5329457 IC50 = 29 nM T80975 CK56SZ 5329458 IC50 = 41 nM T80975 CWZ39N 5329459 IC50 = 1000 nM T80975 CMO84H 5329460 IC50 = 71 nM T80975 CFA21W 5329461 IC50 = 88 nM T80975 CCS62X 5329462 IC50 = 63 nM T80975 CO0VF3 5329463 IC50 = 350 nM T80975 C8NM0W 5329464 IC50 = 265 nM T80975 CY0BN8 5329465 IC50 = 510 nM T80975 C6FOU1 5329466 IC50 = 37 nM T80975 CFS3A4 5329467 IC50 = 24 nM T80975 CKR04W 5329469 IC50 = 14 nM T80975 C9Q1US 5329470 IC50 = 13 nM T80975 CRGY13 5329471 IC50 = 7 nM T80975 C3OE5C 5329472 IC50 = 280 nM T80975 C0U2QK 5329473 IC50 = 28 nM T80975 CLUO27 5329474 IC50 = 41 nM T80975 CYUA16 5329801 IC50 = 5495.41 nM T80975 C19VND 5329802 IC50 > 17000 nM T80975 CI6BY0 5329803 IC50 > 20000 nM T80975 CD0V3Y 5329804 IC50 = 180 nM T80975 C98ZEL 5329806 IC50 = 64.57 nM T80975 CB1DR2 5329807 IC50 = 350 nM T80975 CXS32G 5329808 IC50 = 36 nM T80975 C17MYA 5329812 IC50 = 61.66 nM T80975 CZTJ18 5329814 IC50 = 186 nM T80975 C5CY9J 5329815 IC50 = 57.54 nM T80975 C29BWJ 5329816 IC50 = 18 nM T80975 C0UW5M 5329817 IC50 = 176 nM T80975 CEY86M 5329818 IC50 = 95 nM T80975 C2DA7Q 5329819 IC50 = 117 nM T80975 CCL70T 5329820 IC50 = 269 nM T80975 C7L9NJ 5329821 IC50 = 324 nM T80975 C1FA8H 5329822 IC50 = 5 nM T80975 C52JCD 5329823 IC50 = 35 nM T80975 CX02KO 5329824 IC50 = 2 nM T80975 CJ09MW 5329825 IC50 = 1 nM T80975 CB20GH 5329826 IC50 = 1 nM T80975 CZD5S9 5329827 IC50 = 3 nM T80975 CL7MB8 5329828 IC50 = 6 nM T80975 C35RAQ 5329829 IC50 = 2 nM T80975 CT4L2O 5329830 IC50 = 2 nM T80975 CZFK28 5329831 IC50 = 65 nM T80975 C37HIU 5329832 IC50 = 11 nM T80975 C69MAI 5329833 IC50 = 17 nM T80975 CNF7L0 5329834 IC50 = 26 nM T80975 C0DZ1Y 5329835 IC50 = 29 nM T80975 CRZS03 5329836 IC50 = 31 nM T80975 CH0CJ5 5329837 IC50 = 681 nM T80975 COKV79 5329838 IC50 = 3114 nM T80975 C07MCT 5329839 IC50 = 990 nM T80975 CTR1W9 5329840 IC50 = 4490 nM T80975 CW5L9E 5329841 IC50 = 4 nM T80975 C3CFT6 5329842 IC50 = 150 nM T80975 CL71UW 5329848 IC50 = 720 nM T80975 CW24LT 5329851 IC50 > 10000 nM T80975 CTI5D4 5329853 IC50 = 170 nM T80975 CT3F6Z 5329854 IC50 = 100 nM T80975 CHL9K2 5329855 IC50 = 23 nM T80975 CNX7V5 5329856 IC50 = 50 nM T80975 CB7Z8S 5329857 IC50 = 360 nM T80975 C1TL9F 5329858 IC50 = 22 nM T80975 CKG85D 5329859 IC50 = 141 nM T80975 CWQ0O8 5329860 IC50 = 360 nM T80975 CF4X1J 5329861 IC50 = 93 nM T80975 C8TAE1 5329862 IC50 = 87 nM T80975 C6KDO7 5329863 IC50 = 81 nM T80975 CL46MG 5329864 IC50 = 79 nM T80975 C9T3UE 5329865 IC50 = 51 nM T80975 CYS31K 5329866 IC50 = 18 nM T80975 CQ3B5A 5329867 IC50 = 29 nM T80975 C38MLW 5329868 IC50 = 91 nM T80975 C0ZG9W 5329869 IC50 = 16 nM T80975 CS1VJ5 5329870 IC50 = 15 nM T80975 CCL8O5 5329871 IC50 = 76 nM T80975 CQ8ZH5 5329872 IC50 = 78 nM T80975 C32HVT 5329873 IC50 = 25 nM T80975 C7AZY0 5329874 IC50 = 79 nM T80975 C49TVA 5329875 IC50 = 89 nM T80975 CD0IV1 5329876 IC50 = 39 nM T80975 CE28KH 5329877 IC50 = 1800 nM T80975 CZ64AV 5329878 IC50 > 50000 nM T80975 C29WAO 5329879 IC50 > 50000 nM T80975 CLEQ38 5329880 IC50 = 98 nM T80975 CN5UM6 5329881 IC50 = 1100 nM T80975 CYJ65Z 5329882 IC50 = 19000 nM T80975 CJV8B9 5329883 IC50 = 2100 nM T80975 CM72CQ 5329884 IC50 > 50000 nM T80975 CDI9Z0 5329885 IC50 = 10000 nM T80975 CCMH52 5329886 IC50 = 4400 nM T80975 CO38AK 5329887 IC50 = 430 nM T80975 CCYB15 5329888 IC50 = 7 nM T80975 CUN3E0 5329889 IC50 = 161 nM T80975 CLC18H 5329890 IC50 = 46 nM T80975 C9X4FT 5329891 IC50 = 29 nM T80975 CDQ61V 5329892 IC50 = 520 nM T80975 COY30R 5329893 IC50 = 570 nM T80975 CD98BU 5329894 IC50 = 370 nM T80975 C0N3QG 5329895 IC50 = 50 nM T80975 C17WGL 5329896 IC50 = 83 nM T80975 CV91DU 5329897 IC50 = 39 nM T80975 CBM29R 5329898 IC50 = 23 nM T80975 C3ZSB1 5329899 IC50 = 52 nM T80975 CLPA30 5329900 IC50 = 44 nM T80975 CO9KQ2 5329901 IC50 = 770 nM T80975 CX49RM 5329902 IC50 = 19 nM T80975 CYD94M 5329903 IC50 = 9000 nM T80975 C0ENZ7 5329904 IC50 = 34 nM T80975 CD15LC 5329905 IC50 = 71 nM T80975 C12WJF 5329906 IC50 = 30 nM T80975 C7GEQ6 5329907 IC50 = 6000 nM T80975 CAR8H4 5329908 IC50 > 50000 nM T80975 C2KX0T 5329909 IC50 = 14 nM T80975 C69AGF 5329910 IC50 = 64 nM T80975 CVZ7M0 5329911 IC50 = 470 nM T80975 CTW5N2 5329912 IC50 = 10 nM T80975 C3D0AZ 5329913 IC50 = 350 nM T80975 C23OGR 5329914 IC50 = 21 nM T80975 CP0GB4 5329915 IC50 = 126 nM T80975 CBS40G 5330125 IC50 = 180 nM T80975 CNWK81 5330126 IC50 = 51 nM T80975 CV7GX5 5330127 IC50 = 5 nM T80975 CWAR90 5330128 IC50 = 15 nM T80975 CDG3Z1 5330129 IC50 = 6 nM T80975 C09VSN 5330130 IC50 = 3 nM T80975 CNMJ73 5330131 IC50 = 220 nM T80975 CV4U8Y 5330132 IC50 = 46 nM T80975 C6D7WJ 5330133 IC50 = 6 nM T80975 C2UX4V 5330134 IC50 = 7 nM T80975 CH38FW 5330135 IC50 = 8 nM T80975 CWQ47D 5330136 IC50 = 4 nM T80975 CP2UB6 5330137 IC50 = 2900 nM T80975 CJYX18 5330138 IC50 = 54 nM T80975 CR73WA 5330139 IC50 = 8700 nM T80975 C54VLJ 5330140 IC50 = 3600 nM T80975 C9QO0W 5330141 IC50 = 180 nM T80975 CLD7I9 5330142 IC50 = 1800 nM T80975 CZ8G1N 5330143 IC50 = 110 nM T80975 C7K5PV 5330144 IC50 = 14 nM T80975 CK5CG4 5330145 IC50 = 1200 nM T80975 CPA63S 5330146 IC50 = 130 nM T80975 CY08DW 5330147 IC50 = 25 nM T80975 C6FAS9 5330148 IC50 = 84 nM T80975 CCGA06 5330149 IC50 = 670 nM T80975 C9USJ0 5330150 IC50 = 650 nM T80975 CQX0A3 5330151 IC50 = 1900 nM T80975 CBD8N6 5330152 IC50 = 13000 nM T80975 CX2FO6 5330153 IC50 = 7600 nM T80975 CLI47K 5330157 IC50 = 5 nM T80975 CNI15R 5330158 IC50 = 8 nM T80975 C4IA7N 5330159 IC50 = 6 nM T80975 CSL02W 5330160 IC50 = 15000 nM T80975 CNA8R7 5330161 IC50 = 1400 nM T80975 CF4JU8 5330162 IC50 = 55000 nM T80975 CDY0R5 5330163 IC50 = 6600 nM T80975 CR0GX9 5330164 IC50 = 10000 nM T80975 C37DGR 5330165 IC50 = 20000 nM T80975 CW8G9J 5330166 IC50 = 62 nM T80975 C7Z2YH 5330167 IC50 = 21 nM T80975 CEX9A7 5330168 IC50 = 190 nM T80975 C3I6KF 5330169 IC50 = 71 nM T80975 CY7K6I 5330170 IC50 = 1110 nM T80975 CI32HV 5330173 IC50 = 1180 nM T80975 C7Y2VN 5330175 IC50 = 670 nM T80975 C3Q1SK 5330176 IC50 = 250 nM T80975 CC4Z9K 5330178 IC50 = 1230 nM T80975 C2H1EQ 5330179 IC50 = 410 nM T80975 C04DHT 5330180 IC50 = 1380 nM T80975 COF57G 5330182 IC50 = 100 nM T80975 CH9SZ3 5330184 IC50 = 420 nM T80975 CA09XJ 5330186 IC50 = 2320 nM T80975 CA5H0W 5330187 IC50 = 4960 nM T80975 C5RK3H 5330188 IC50 = 17030 nM T80975 C6NMP8 5330189 IC50 = 42640 nM T80975 CW81JE 5330190 IC50 = 8160 nM T80975 CQDI38 5330194 IC50 = 91350 nM T80975 CUZ0I1 5330195 IC50 = 73820 nM T80975 CD7U5B 5330196 IC50 = 15600 nM T80975 CB23PA 5330197 IC50 = 2170 nM T80975 C6BPR5 5330198 IC50 = 77000 nM T80975 C7USC4 5330359 IC50 = 168 nM T80975 CU7VS2 5330360 IC50 = 740 nM T80975 CC7HB9 5330361 IC50 = 1010 nM T80975 C30QCV 5330362 IC50 = 76 nM T80975 C6QCZ0 5330363 IC50 = 1000 nM T80975 CT5IB7 5330364 IC50 = 189 nM T80975 CKF4G9 5330365 IC50 = 1047.13 nM T80975 CT01YE 5330366 IC50 > 10000 nM T80975 CWLU89 5330367 IC50 = 1600 nM T80975 CSG61Y 5330368 IC50 = 275 nM T80975 CQZ06G 5330369 IC50 = 134.9 nM T80975 CGPM14 5330370 IC50 = 4265.8 nM T80975 CNGW06 5330371 IC50 = 2380 nM T80975 C0OV7Q 5330372 IC50 = 346 nM T80975 CV74KI 5330373 IC50 = 302 nM T80975 CZEN87 5330374 IC50 = 588.84 nM T80975 CH0C7O 5330375 IC50 > 10000 nM T80975 CPJU86 5330376 IC50 > 10000 nM T80975 CE9R0A 5330377 IC50 > 10000 nM T80975 C7J9XO 5330378 IC50 = 234.42 nM T80975 CS94FE 5330379 IC50 = 123 nM T80975 CFK2I3 5330380 IC50 = 181.97 nM T80975 CYJ9M5 5330381 IC50 = 399 nM T80975 CAT79J 5330382 IC50 = 391 nM T80975 CP26UZ 5330383 IC50 = 263.03 nM T80975 C25CEU 5330384 IC50 = 2290.87 nM T80975 CK16CV 5330385 IC50 > 10000 nM T80975 C9RE5L 5330386 IC50 = 568 nM T80975 CZ3LK2 5330387 IC50 = 84 nM T80975 CRU94N 5330388 IC50 = 63 nM T80975 CDB68F 5330389 IC50 = 105 nM T80975 C7CX0H 5330390 IC50 = 75.86 nM T80975 C8E0XS 5330391 IC50 = 93.33 nM T80975 CW1VX9 5330392 IC50 = 67.61 nM T80975 C4A3GV 5330393 IC50 = 610 nM T80975 CGV36U 5330394 IC50 = 251 nM T80975 CAD7N3 5330395 IC50 > 10000 nM T80975 CU7VK6 5330396 IC50 = 1348.96 nM T80975 CW2MT7 5330397 IC50 > 10000 nM T80975 CH7XF6 5330398 IC50 > 10000 nM T80975 C9ACY8 5330399 IC50 > 10000 nM T80975 CR1CV4 5330401 IC50 = 497 nM T80975 CSD47J 5330402 IC50 > 10000 nM T80975 C58VWF 5330403 IC50 = 500 nM T80975 CXP8M2 5330404 IC50 = 761 nM T80975 CGE78Y 5330405 IC50 > 10000 nM T80975 C7E4HZ 5330406 IC50 = 708 nM T80975 CA7U4J 5330407 IC50 = 2110 nM T80975 CF01JS 5330804 IC50 = 51 nM T80975 C3U0TG 5330830 IC50 > 100000 nM T80975 CL1FH5 5330832 IC50 > 100000 nM T80975 C1P2ZA 5330847 IC50 > 100000 nM T80975 CS3A8F 5331081 IC50 > 20000 nM T80975 CG4W8K 5331082 IC50 = 6600 nM T80975 CD4C2A 5331083 IC50 = 6600 nM T80975 C6AT8V 5331084 IC50 = 6700 nM T80975 CJVS23 5331085 IC50 > 20000 nM T80975 CZ29FN 5331086 IC50 = 6200 nM T80975 CYL78A 5331087 IC50 = 10000 nM T80975 CJ87XR 5331088 IC50 > 20000 nM T80975 CFB3K7 5331089 IC50 = 11000 nM T80975 C9WY1O 5331090 IC50 > 20000 nM T80975 C9ZK3D 5331091 IC50 = 1200 nM T80975 C6RJC8 5331092 IC50 = 490 nM T80975 C0IOY8 5331093 IC50 > 20000 nM T80975 CMD08O 5331094 IC50 = 2000 nM T80975 C87VQB 5353854 IC50 = 390 nM T80975 CDQ3M7 5359485 IC50 = 0.92 ug.mL-1 T80975 C54BYP 5360741 IC50 = 1.1 ug.mL-1 T80975 C2O9ZG 5391486 IC50 = 9610 nM T80975 C15RJZ 5398217 IC50 = 9600 nM T80975 CCT39K 5703472 IC50 = 1130 nM T80975 CDK3J0 5703619 IC50 = 7.7 nM T80975 C2DCW3 5916724 IC50 = 7000 nM T80975 CAI5Y2 5941539 IC50 = 700 nM T80975 CEZP52 6263849 IC50 > 50000 nM T80975 C6Y5HN 6312547 IC50 = 20000 nM T80975 CV2KQ1 6326407 IC50 = 4 nM T80975 CF46XV 6326408 IC50 = 10 nM T80975 C2H3UZ 6326413 IC50 = 3500 nM T80975 C49DUV 6326414 IC50 = 1600 nM T80975 C7ZB6K 6326415 IC50 = 1300 nM T80975 CJN34Y 6326416 IC50 > 10000 nM T80975 C9WDE8 6326417 IC50 > 10000 nM T80975 C1P5HD 6326418 IC50 = 410 nM T80975 CDWI70 6326419 IC50 = 240 nM T80975 CZJ1R9 6326420 IC50 > 10000 nM T80975 CPO78D 6326421 IC50 = 4700 nM T80975 CBD49X 6326422 IC50 = 210 nM T80975 CSXG59 6406980 IC50 > 10000 nM T80975 C08LWD 6406981 IC50 > 10000 nM T80975 CM80PH 6407032 IC50 > 10000 nM T80975 CSN2K0 6407119 IC50 > 10000 nM T80975 CB84OI 6407141 IC50 > 10000 nM T80975 C0IYS8 6408948 IC50 = 7.3 nM T80975 CN0M7W 6411110 IC50 = 1.6 nM T80975 C7Z4JC 6411759 IC50 > 10000 nM T80975 C0E6RD 6413680 IC50 = 360 nM T80975 C18VEH 6415635 IC50 = 6.2 nM T80975 C53UGK 6419378 IC50 = 650 nM T80975 CK3A1M 6419379 IC50 = 4700 nM T80975 C1Y8LP 6419380 IC50 = 1700 nM T80975 C3DO7L 6419381 IC50 = 1400 nM T80975 CJ6QB4 6419382 IC50 = 610 nM T80975 CQO68G 6419383 IC50 = 130 nM T80975 CV5C7R 6419384 IC50 > 10000 nM T80975 C27ZIA 6419385 IC50 = 870 nM T80975 C6L5HS 6419386 IC50 = 950 nM T80975 C3CQW0 6419387 IC50 = 80 nM T80975 CWOA63 6419388 IC50 = 210 nM T80975 CZVU64 6419389 IC50 = 200 nM T80975 C9FN4B 6419390 IC50 = 240 nM T80975 CN53YW 6419391 IC50 = 670 nM T80975 C17NWJ 6419392 IC50 = 30 nM T80975 C13IRC 6419393 IC50 = 140 nM T80975 C4FLE9 6419394 IC50 = 40 nM T80975 C4GHT0 6419395 IC50 = 300 nM T80975 C8SAQ1 6419396 IC50 = 380 nM T80975 CP71CL 6419397 IC50 = 200 nM T80975 CSMU27 6425419 Ki = 0.2 nM T80975 C2N0IR 6477203 IC50 = 10300 nM T80975 CYP69H 6482470 IC50 = 2000 nM T80975 CNFV70 6539738 IC50 > 48000 nM T80975 CBRC53 6539739 IC50 > 47000 nM T80975 C8QG1T 6539740 IC50 > 48000 nM T80975 CW7VD6 6539741 IC50 = 3550 nM T80975 C5UFS1 6539742 IC50 = 1020 nM T80975 C5XSJ6 6539743 IC50 > 48000 nM T80975 CRL2P4 6539744 IC50 > 48000 nM T80975 CSWR78 6539745 IC50 > 48000 nM T80975 CXI8M7 6539746 IC50 = 12300 nM T80975 CSZF21 6539747 IC50 = 21900 nM T80975 CFM2K9 6539748 IC50 > 48000 nM T80975 C1QFC6 6539749 IC50 = 830 nM T80975 CFQ5R7 6539750 IC50 = 2040 nM T80975 C0R6WV 6539751 IC50 = 630 nM T80975 C25FMB 6539752 IC50 = 2040 nM T80975 CRB1O3 6539753 IC50 = 3240 nM T80975 CZ17AH 6539754 IC50 > 23000 nM T80975 CT4K0Z 6539755 IC50 > 20000 nM T80975 CMIS20 6539756 IC50 > 20000 nM T80975 CTNR52 6539757 IC50 > 19000 nM T80975 CJ58QK 6539758 IC50 > 24000 nM T80975 CA31PJ 6539953 IC50 = 5320 nM T80975 C64ZJA 6539954 IC50 = 3810 nM T80975 CBD1H7 6539955 IC50 > 50000 nM T80975 CWHY29 6539956 IC50 > 50000 nM T80975 CW76RA 6539957 IC50 = 34000 nM T80975 C7K1QS 6539958 IC50 = 263 nM T80975 CJ7IL2 6539959 IC50 > 50000 nM T80975 CH86XJ 6539961 IC50 > 50000 nM T80975 C41FUH 6539962 IC50 > 50000 nM T80975 C7M2JP 6539963 IC50 > 50000 nM T80975 CS5V1C 6539964 IC50 = 34600 nM T80975 C10FYS 6539966 IC50 > 50000 nM T80975 CIS1T3 6539967 IC50 = 435 nM T80975 CUFE90 6539968 IC50 = 4600 nM T80975 C5FD7G 6539969 IC50 = 4570.88 nM T80975 C15HWY 6539970 IC50 > 50000 nM T80975 CTZ4W0 6539971 IC50 = 10 nM T80975 CAOU70 6539972 IC50 = 6.026 nM T80975 C8A7ZI 6539973 IC50 > 50000 nM T80975 C3VW9T 6539974 IC50 = 2818.38 nM T80975 C6Z0AQ 6539975 IC50 = 1096.48 nM T80975 C7TK3A 6539976 IC50 > 50000 nM T80975 C2BRQ3 6539977 IC50 = 170 nM T80975 CEM48C 6539978 IC50 = 758.58 nM T80975 CIM45N 6539979 IC50 = 54.95 nM T80975 CQU47G 6539980 IC50 = 1905.46 nM T80975 C5NF1H 6539981 IC50 = 330 nM T80975 CBA9I6 6539982 IC50 = 790 nM T80975 CE9L8Y 6539983 IC50 = 26.3 nM T80975 C0RH8N 6539984 IC50 = 169.82 nM T80975 CUPQ08 6539985 IC50 = 1 nM T80975 C24QDV 6539986 IC50 = 181.97 nM T80975 C90DZT 6539987 IC50 = 1698.24 nM T80975 CK9TD3 6539988 IC50 = 257.04 nM T80975 CDA25S 6539989 IC50 = 52.48 nM T80975 C6Q4ZY 6539990 IC50 = 109.65 nM T80975 C3SXL8 6539991 IC50 = 34.67 nM T80975 CWC68D 6539992 IC50 = 69 nM T80975 CR9GL1 6539993 IC50 = 109.65 nM T80975 CK23SV 6539994 IC50 = 54.95 nM T80975 C9ZN6H 6539995 IC50 = 52 nM T80975 C39QGE 6539996 IC50 = 338.84 nM T80975 C8EJI1 6539997 IC50 = 34.67 nM T80975 CYQ9D4 6539998 IC50 = 95.5 nM T80975 CH2EV5 6539999 IC50 = 45.71 nM T80975 C9GMT4 6540000 IC50 = 120.23 nM T80975 CWA5M6 6540001 IC50 = 10 nM T80975 C3SAD6 6540002 IC50 = 295.12 nM T80975 CU14NK 6540003 IC50 = 12 nM T80975 CIC64F 6540004 IC50 = 158.49 nM T80975 CMEZ23 6540005 IC50 = 45 nM T80975 CG1L6R 6540006 IC50 = 16.98 nM T80975 C92OFS 6540007 IC50 = 330 nM T80975 C7H4QP 6540008 IC50 = 210 nM T80975 CF97JX 6540009 IC50 = 210 nM T80975 C52OIP 6540010 IC50 = 588.84 nM T80975 C81QDX 6540011 IC50 = 180 nM T80975 C2O4MX 6540012 IC50 = 26 nM T80975 C6HWM9 6540013 IC50 = 128.82 nM T80975 CB9N7T 6540014 IC50 = 280 nM T80975 CSGQ06 6540015 IC50 = 34 nM T80975 CP32OT 6540016 IC50 = 52.48 nM T80975 C4NWO7 6540017 IC50 = 19 nM T80975 C8AU3M 6540018 IC50 = 64 nM T80975 C3K7TM 6540019 IC50 = 15 nM T80975 CM1TH0 6540020 IC50 = 229.09 nM T80975 CK19HQ 6540021 IC50 = 10.96 nM T80975 CXK07R 6540022 IC50 = 100 nM T80975 CFLH24 6540023 IC50 = 100 nM T80975 CJ17TA 6540024 IC50 = 19 nM T80975 C0BQ2E 6540025 IC50 = 83.18 nM T80975 CIUP42 6540026 IC50 = 12.88 nM T80975 C0PUR2 6540027 IC50 = 151.36 nM T80975 CE7A5Z 6540028 IC50 = 50.12 nM T80975 C8U9HT 6540029 IC50 = 3.02 nM T80975 CP0XI6 6603792 IC50 = 1570 nM T80975 C5OG3Q 6625323 IC50 = 4.1 nM T80975 CG17TN 6914611 IC50 > 50000 nM T80975 C7E2QK 6914613 IC50 > 50000 nM T80975 CVU8N0 6918710 IC50 > 20000 nM T80975 C14UAT 7574840 IC50 > 10000 nM T80975 CV7L5M 8895911 IC50 > 10000 nM T80975 CY2R3K 9124858 IC50 = 3.4 nM T80975 C4G9WR 9547398 IC50 > 100000 nM T80975 C76CUP 9547698 IC50 = 4600 nM T80975 C4A8RX 9794758 IC50 = 1440 nM T80975 CK21EQ 9796713 IC50 = 110 nM T80975 CL34UJ 9799758 IC50 = 71 nM T80975 CI80BK 9803350 IC50 = 2700 nM T80975 C0B8AY 9818223 IC50 = 10 nM T80975 C5B1NS 9822610 IC50 = 6.3 nM T80975 C1E2DV 9826083 IC50 > 10000 nM T80975 C9TAL6 9826308 IC50 = 360 nM T80975 CFH1J9 9839988 IC50 = 100 nM T80975 CJH69P 9840393 IC50 > 300 nM T80975 CKL02D 9847304 IC50 = 76 nM T80975 C41QWA 9857146 IC50 > 10000 nM T80975 C43FVO 9859850 IC50 = 60 nM T80975 CY9T2V 9862137 IC50 = 49 nM T80975 C16VXB 9863538 IC50 = 3500 nM T80975 CRC65X 9863786 IC50 > 10000 nM T80975 CRU2S7 9864300 Ki = 17 nM T80975 CW8V0K 9864418 IC50 > 20000 nM T80975 C5YF4Z 9870238 IC50 = 32 nM T80975 CG4U2Q 9881010 Ki > 10000 nM T80975 C9LE7U 9883063 IC50 = 46 nM T80975 CE47IF 9884465 IC50 = 80 nM T80975 C18HKQ 9885748 IC50 = 770 nM T80975 C4LD6H 9888708 IC50 = 4 nM T80975 CHF7G5 9890746 IC50 = 17300 nM T80975 CXA5C8 9893493 IC50 = 0.062 nM T80975 CT1EK0 9902148 Ki = 106 nM T80975 C54KXJ 9903480 IC50 > 10000 nM T80975 C7BEL6 9906150 IC50 = 200 nM T80975 C5BSO0 9908026 IC50 = 69 nM T80975 C2TC1L 9910609 IC50 = 12 nM T80975 CFA49P 9910872 IC50 = 26 nM T80975 C3EUB4 9911005 IC50 > 100000 nM T80975 CRO5D3 9912410 IC50 = 19 nM T80975 CQY1L2 9924662 Ki > 10000 nM T80975 CX23IZ 9926213 IC50 > 10000 nM T80975 CTQ48P 9927432 IC50 = 186 nM T80975 CYW49X 9927718 IC50 > 25000 nM T80975 C1BZ0P 9928737 IC50 = 5 nM T80975 CQ64LI 9935852 IC50 = 3.5 nM T80975 CP2S5A 9936664 IC50 = 16 nM T80975 CS5KX9 9938299 IC50 = 4.2 nM T80975 CZXI68 9944849 Ki = 320 nM T80975 CB8L3A 9948660 IC50 = 24 nM T80975 C30KCV 9950381 IC50 = 32 nM T80975 C54ZXH 9950678 IC50 = 2290 nM T80975 CD5M3J 9952008 IC50 = 40 nM T80975 C5LA8Y 9958299 IC50 = 3.3 nM T80975 C3P0XT 9968566 IC50 = 450 nM T80975 C0WQT7 9968862 Ki = 19 nM T80975 CNX36L 9970036 Ki = 91 nM T80975 CSRU93 9975630 IC50 > 10000 nM T80975 CHB0D2 9982235 IC50 = 11 nM T80975 C37GXK 9983303 IC50 > 20000 nM T80975 CCJ93T 9999811 IC50 = 4140 nM T80975 C26QHZ 10005638 IC50 > 10000 nM T80975 CR8DA1 10024683 IC50 > 100000 nM T80975 C7CR9Q 10025788 IC50 = 225 nM T80975 CBF3T6 10043847 IC50 = 2010 nM T80975 CG57EC 10047098 IC50 = 49900 nM T80975 CLA93G 10047202 IC50 = 4850 nM T80975 C3LCH5 10047545 IC50 > 100000 nM T80975 C7YD1X 10048045 IC50 > 25000 nM T80975 CUJR40 10062694 EC50 = 22 nM T80975 CH31FR 10067064 IC50 = 100 nM T80975 C1JUF8 10073832 IC50 = 57 nM T80975 C2C1BP 10089048 IC50 > 20000 nM T80975 C74VKR 10111613 IC50 = 12 nM T80975 CY28QV 10113430 IC50 > 2000 nM T80975 CIV15Q 10113978 IC50 = 30 nM T80975 CUC8F7 10115116 IC50 = 411 nM T80975 CWC0K6 10115117 IC50 = 18 nM T80975 C0Q3CB 10116002 IC50 = 130 nM T80975 CV67EI 10117977 IC50 = 3.4 nM T80975 CT96JK 10120050 IC50 = 16.5 nM T80975 CTXW95 10126509 IC50 = 400 nM T80975 CA31MX 10131256 IC50 = 400 nM T80975 CK34VR 10131963 Ki = 2 nM T80975 CC34SL 10137291 IC50 = 73 nM T80975 CR3U0X 10138086 Ki = 38 nM T80975 CPMD80 10140205 IC50 = 309 nM T80975 C3JGH7 10141033 IC50 = 2.6 nM T80975 CNRX37 10142514 IC50 = 26 nM T80975 CDTB71 10151417 IC50 = 25 nM T80975 CREM37 10151881 IC50 = 480 nM T80975 C69DHW 10158652 IC50 < 16000 nM T80975 C9ILB7 10160584 IC50 = 21 nM T80975 C3FGO2 10160775 IC50 = 2.9 nM T80975 CIQG50 10161259 IC50 = 7.6 nM T80975 C3TZ1Y 10163749 IC50 = 1.1 nM T80975 C29JTQ 10164190 IC50 = 2.3 nM T80975 C7X6KB 10165834 IC50 = 40 nM T80975 C1Q6OJ 10166498 IC50 = 5.4 nM T80975 C8YZL0 10171618 IC50 = 3200 nM T80975 CC78NE 10179293 IC50 = 94 nM T80975 C67IQW 10180253 Ki = 490 nM T80975 C67PWJ 10181898 IC50 = 21500 nM T80975 CDZX43 10182654 IC50 = 12 nM T80975 C7GN8Q 10183216 IC50 = 5.4 nM T80975 CU0WT6 10184615 IC50 = 5 nM T80975 CJU67H 10186182 IC50 = 27 nM T80975 CZI8M7 10186183 IC50 = 420 nM T80975 C1KNM3 10186269 IC50 = 10 nM T80975 CNAR49 10198951 IC50 = 320 nM T80975 C1TX8D 10198953 IC50 > 10000 nM T80975 C2RLF5 10199254 IC50 = 20 nM T80975 CL49QV 10199918 IC50 = 55 nM T80975 C0C8OQ 10200879 IC50 = 208 nM T80975 CCXY21 10204357 IC50 = 6.3 nM T80975 CGOT91 10207821 IC50 = 1410 nM T80975 C8B0CW 10207842 IC50 > 10000 nM T80975 C0D3XA 10209627 IC50 = 1000 nM T80975 C7MVB8 10214675 IC50 > 20000 nM T80975 C5V6PK 10216157 IC50 = 63 nM T80975 CE2G4B 10216381 IC50 = 63 nM T80975 CEW30I 10217590 IC50 > 10000 nM T80975 C4HQB1 10223401 IC50 = 17 nM T80975 C62MDP 10225270 IC50 = 65 nM T80975 C1RGN4 10226262 IC50 = 57 nM T80975 CPE29J 10229538 IC50 = 50 nM T80975 C1VUP6 10229632 IC50 = 1.3 nM T80975 CZX26W 10230568 IC50 = 5.1 nM T80975 CF90MC 10230609 IC50 = 4000 nM T80975 CD7J3O 10231458 IC50 > 30000 nM T80975 C1A5HT 10233129 IC50 = 38 nM T80975 C8HN7C 10246119 IC50 > 50000 nM T80975 CC9E5Q 10249989 IC50 = 40 nM T80975 C1WL8B 10251852 IC50 = 132100 nM T80975 CH30RC 10253133 IC50 > 10000 nM T80975 CS46QO 10269041 IC50 = 1400 nM T80975 C7BL5I 10273106 IC50 = 111 nM T80975 C2EO1A 10273854 IC50 = 17 nM T80975 CFE0U6 10275000 IC50 = 13 nM T80975 C6DC8Q 10275163 IC50 = 1100 nM T80975 C2F6DJ 10275349 IC50 = 15 nM T80975 CJGH26 10275985 IC50 = 1370 nM T80975 C5HC0D 10276395 IC50 = 603 nM T80975 C12YUR 10278843 IC50 = 16 nM T80975 C60ZOC 10278844 IC50 = 5.4 nM T80975 CTHI58 10279624 IC50 = 2.1 nM T80975 CW8OB2 10279981 IC50 = 400 nM T80975 C10UBJ 10280848 IC50 > 20000 nM T80975 CDG1X4 10286382 IC50 = 2500 nM T80975 CGN04D 10288960 IC50 = 30 nM T80975 CD0W7J 10290951 Ki = 8 nM T80975 CT84CH 10291174 Ki = 120 nM T80975 CC82SP 10293612 Ki = 23 nM T80975 C7YK8W 10295715 Ki = 70 nM T80975 C7SFI1 10296883 IC50 = 3900 nM T80975 CVO54Z 10300451 IC50 > 20000 nM T80975 CFY14M 10300768 IC50 = 17 nM T80975 C8RD3V 10301884 IC50 = 2500 nM T80975 CAM42B 10301885 IC50 = 2000 nM T80975 CP1LO7 10302209 IC50 = 9500 nM T80975 CRAB41 10317147 IC50 = 1067 nM T80975 CIK4R9 10319429 IC50 = 120 nM T80975 C5CBF9 10320381 IC50 = 500 nM T80975 C7OA9P 10325135 IC50 = 79 nM T80975 CTX01B 10341351 IC50 = 5030 nM T80975 C9ZXG2 10357919 IC50 = 84000 nM T80975 CT9B4R 10362034 IC50 = 24 nM T80975 CNK0W6 10386095 IC50 = 130 nM T80975 C07XHY 10388612 IC50 = 8 nM T80975 CQ6OF5 10388672 IC50 = 110 nM T80975 CA8B5T 10390073 IC50 = 1700 nM T80975 C4G2EI 10409523 IC50 = 170 nM T80975 C5ZD3T 10409591 IC50 = 79 nM T80975 CLAX64 10413508 IC50 = 2600 nM T80975 C4CP7K 10423452 IC50 = 800 nM T80975 CY9F3G 10425574 IC50 = 0.6 nM T80975 C7HBP6 10429593 IC50 > 10000 nM T80975 CV2N0G 10431226 Ki > 6660 nM T80975 CFLH53 10432113 IC50 > 1000 nM T80975 C2VPT6 10436729 IC50 = 16 nM T80975 C3FT4K 10450827 IC50 = 46 nM T80975 CL7PF2 10451087 IC50 = 3600 nM T80975 C95LYF 10457505 IC50 > 100000 nM T80975 C4CV5L 10470475 IC50 = 10000 nM T80975 CH4CY9 10471016 IC50 = 600 nM T80975 C7PLI5 10478569 IC50 = 18 nM T80975 CRX6F0 10479082 IC50 > 20000 nM T80975 CJ5M1D 10482445 IC50 = 400 nM T80975 CEML49 10538870 IC50 = 35000 nM T80975 C9O2PG 10588346 IC50 = 3000 nM T80975 C7KF2E 10705154 IC50 = 3000 nM T80975 C83QWV 10714343 IC50 = 4810 nM T80975 C4D5LN 10717065 Ki = 0.4 nM T80975 C2C8GH 10732141 IC50 = 9000 nM T80975 CJ4P5T 10905857 IC50 > 100000 nM T80975 CDE08I 11140977 Ki = 25000 nM T80975 C2ND0F 11149670 Ki = 8 nM T80975 CPC3S4 11150615 IC50 = 8000 nM T80975 C03XHM 11152545 IC50 = 16 nM T80975 CT9DB1 11154117 IC50 = 187 nM T80975 CW6Z5P 11154134 IC50 = 9 nM T80975 CR2O3F 11155047 IC50 = 70 nM T80975 COMB49 11155938 IC50 = 17 nM T80975 C84NJO 11155950 IC50 = 6 nM T80975 CB47NS 11156401 IC50 = 22 nM T80975 CQ73KF 11156617 IC50 = 0.5 nM T80975 C8L0AV 11156649 Ki = 10 nM T80975 CQ1A2U 11156873 Ki = 2 nM T80975 CUT50K 11156969 Ki = 10 nM T80975 CIA1Q6 11167070 IC50 = 5.6 nM T80975 CXC91Z 11167118 Ki = 9 nM T80975 C3K6ST 11167612 IC50 = 2 nM T80975 C7V8JR 11167666 IC50 = 66 nM T80975 CN2JQ0 11169051 IC50 > 25000 nM T80975 C6KMU2 11176194 IC50 = 23 nM T80975 CU53KH 11177394 IC50 = 6161 nM T80975 C7ZB5L 11177668 IC50 = 36 nM T80975 CNG8F1 11178869 IC50 = 1200 nM T80975 C2BQD8 11179315 Ki = 2 nM T80975 C05MCD 11188653 IC50 = 105 nM T80975 CD9E2W 11188787 IC50 = 96 nM T80975 C6H5VA 11189551 IC50 = 42 nM T80975 C5IM3N 11190081 Ki = 8 nM T80975 CX0QO7 11192412 IC50 = 25 nM T80975 C0Y8TX 11192751 IC50 = 480 nM T80975 CEUR60 11192985 IC50 = 3300 nM T80975 C58BGW 11197220 IC50 = 400 nM T80975 COK51D 11202270 IC50 = 190 nM T80975 CB06ZF 11204217 IC50 = 5500 nM T80975 CJNS72 11209305 IC50 = 320 nM T80975 C8G5WP 11210533 IC50 = 390 nM T80975 C8T2NG 11211389 IC50 = 1.3 nM T80975 CP4GL8 11212549 IC50 = 0.2 nM T80975 CT7X1E 11213083 IC50 = 0.2 nM T80975 CT3K9Z 11213588 IC50 = 1 nM T80975 C5F2PA 11213751 IC50 = 8 nM T80975 CG29JX 11214363 IC50 = 11 nM T80975 CEJ6F2 11214762 IC50 = 4200 nM T80975 CF2GE5 11222252 IC50 = 1000 nM T80975 CSWR60 11223082 IC50 = 628 nM T80975 CB0MO3 11223754 IC50 = 34 nM T80975 CWC2X6 11223992 IC50 = 76 nM T80975 CY2PF1 11224592 IC50 = 0.2 nM T80975 CQ4XT3 11224593 IC50 = 22 nM T80975 C06FWR 11224992 IC50 = 5.9 nM T80975 C7Q2TJ 11225298 IC50 = 270 nM T80975 CW94ZU 11225456 IC50 = 5.6 nM T80975 C9CGI8 11225457 IC50 = 37 nM T80975 CAG8J0 11225774 IC50 = 1 nM T80975 CE6T8H 11231939 IC50 = 380 nM T80975 C2W5RC 11235063 IC50 > 30000 nM T80975 CT0C5R 11235290 IC50 = 37 nM T80975 CFJ0W9 11236257 IC50 > 100 nM T80975 CFJ2C0 11236308 IC50 = 1.8 nM T80975 C8S2HR 11237059 IC50 = 27 nM T80975 CVOW82 11238420 IC50 > 50000 nM T80975 C04KZE 11242074 Ki = 530 nM T80975 CICX97 11244488 IC50 = 140 nM T80975 C8CF1H 11244819 IC50 = 64 nM T80975 C1Y7DB 11245809 IC50 = 5 nM T80975 C4R2CE 11247801 IC50 < 1 nM T80975 C8GP7B 11248025 IC50 = 19 nM T80975 C2GXU7 11248659 Ki = 4 nM T80975 C61NBY 11248850 IC50 = 2 nM T80975 C30PKR 11248978 IC50 > 20000 nM T80975 C8JIV1 11253284 Ki = 818 nM T80975 CD9T6R 11257328 IC50 = 11 nM T80975 C8DHX0 11257497 IC50 = 250 nM T80975 CRZW58 11258149 IC50 > 10000 nM T80975 CJFX60 11259128 IC50 = 10 nM T80975 C71ONE 11259460 IC50 = 1.6 nM T80975 COW4I8 11259499 IC50 = 4 nM T80975 CLE31R 11259708 IC50 = 1.1 nM T80975 CV18PX 11265647 IC50 = 12500 nM T80975 CJ23CR 11268446 IC50 = 21 nM T80975 CBQ10L 11268741 IC50 = 6 nM T80975 CPI45C 11270447 IC50 = 0.4 nM T80975 CNBX16 11270660 IC50 > 10000 nM T80975 CMZ49B 11270888 IC50 = 0.7 nM T80975 CQL3P9 11271710 IC50 = 21 nM T80975 CEP0G1 11273105 IC50 = 530 nM T80975 CI1H5P 11280431 IC50 = 67 nM T80975 C3QKJ0 11281671 IC50 = 11 nM T80975 CC24PZ 11281789 IC50 = 247 nM T80975 C6C3JX 11281930 IC50 = 1900 nM T80975 CE6HF7 11282447 IC50 = 11 nM T80975 CUO27S 11282791 IC50 < 1 nM T80975 C0WY4J 11283899 Ki = 3 nM T80975 C8FGR1 11288910 IC50 > 2000 nM T80975 C27TCQ 11289252 Ki = 0.47 nM T80975 CO69LG 11289317 Ki = 0.28 nM T80975 CC9OM5 11292923 IC50 = 0.2 nM T80975 CBOP58 11293798 Ki > 8210 nM T80975 C2IA4K 11294266 IC50 = 1 nM T80975 CSXY78 11294864 IC50 > 20000 nM T80975 C9S8PK 11295293 IC50 > 25000 nM T80975 C60ISR 11304968 IC50 = 80 nM T80975 CHKY86 11305057 IC50 = 0.5 nM T80975 C8CL6Y 11305897 IC50 = 276 nM T80975 CP4KA1 11307497 Ki = 0.2 nM T80975 CU3S9G 11311349 IC50 = 500 nM T80975 CYK15J 11314310 IC50 = 13 nM T80975 CHQ6O9 11316725 IC50 > 100 nM T80975 CGMD57 11316827 IC50 = 66 nM T80975 CPU9I3 11316975 IC50 > 20000 nM T80975 CLX54H 11317348 IC50 = 0.9 nM T80975 C3YA8L 11318315 IC50 = 36 nM T80975 CL7G8F 11325920 IC50 = 23 nM T80975 C6S7VQ 11326107 IC50 = 48 nM T80975 CI75ZE 11327388 IC50 = 32 nM T80975 C2MY9F 11327849 IC50 = 2.3 nM T80975 CC8J3N 11328182 IC50 = 71 nM T80975 C9GI6J 11328439 IC50 = 0.7 nM T80975 CGP80V 11328586 IC50 = 1 nM T80975 CQ8I4H 11328863 IC50 > 20000 nM T80975 CBZS09 11329617 IC50 = 0.7 nM T80975 CU5P8C 11331007 IC50 = 5000 nM T80975 CY54IT 11337407 IC50 = 497 nM T80975 CK1P7Y 11337894 IC50 = 8 nM T80975 C9BZ5Q 11339914 IC50 = 0.4 nM T80975 C4VB3D 11339915 IC50 = 1.1 nM T80975 CL6WN0 11340353 IC50 = 2 nM T80975 CUT16W 11340683 IC50 = 25 nM T80975 C40AXU 11341153 Ki = 3 nM T80975 CWR1D2 11346327 IC50 = 1000 nM T80975 CPKO20 11350036 IC50 = 270 nM T80975 CIR2X8 11350984 IC50 = 13 nM T80975 CI6ZX5 11350985 IC50 = 1.2 nM T80975 CEC31B 11351900 IC50 = 0.1995 nM T80975 CA6F4L 11352215 IC50 = 23 nM T80975 C12LUM 11352232 IC50 = 0.4 nM T80975 CL56UQ 11352732 Ki = 5 nM T80975 CDZR14 11357877 IC50 > 10000 nM T80975 CRTG16 11359538 IC50 = 500 nM T80975 C26BZX 11362471 Ki > 8210 nM T80975 CB45PJ 11362483 IC50 = 12 nM T80975 CRN59I 11363357 IC50 = 2 nM T80975 CMNS96 11363515 IC50 = 1200 nM T80975 CT86QF 11363728 IC50 = 3 nM T80975 C9B4XP 11363872 IC50 = 1 nM T80975 CGN8P2 11365768 IC50 = 4000 nM T80975 CY8AQ4 11371508 IC50 = 15 nM T80975 CMN14Z 11373591 IC50 = 5 nM T80975 C43NPS 11373886 IC50 > 10000 nM T80975 C25ZCN 11374110 IC50 = 11 nM T80975 CL4Z7M 11374372 IC50 = 1.8 nM T80975 CG57WD 11374515 IC50 = 17 nM T80975 CJ75ZF 11375010 IC50 = 4 nM T80975 CP4ZO0 11375301 IC50 = 0.5012 nM T80975 CT6Y9W 11376799 IC50 = 7400 nM T80975 C6L9HV 11380352 Ki = 0.13 nM T80975 C4H0ZP 11380375 IC50 > 2000 nM T80975 C4IH5E 11383525 IC50 = 0.45 nM T80975 C0S1OV 11385268 IC50 = 1.1 nM T80975 C05CWH 11392350 IC50 = 930 nM T80975 C6PW4B 11394942 IC50 = 163 nM T80975 CY8QP1 11396878 IC50 = 12 nM T80975 CWXB93 11397177 Ki > 8210 nM T80975 CT3VP7 11398307 IC50 = 1 nM T80975 CEV1O4 11398610 IC50 = 933 nM T80975 CNT8W2 11404903 IC50 = 153 nM T80975 CPIM91 11406239 IC50 = 13 nM T80975 C6EP7S 11407183 IC50 = 8 nM T80975 CL7I5H 11407736 IC50 = 90 nM T80975 CX25IH 11407794 IC50 = 15 nM T80975 C4GTW1 11408569 IC50 = 350 nM T80975 CJUC63 11409093 IC50 = 8.9 nM T80975 CL1FN7 11409568 IC50 = 3 nM T80975 C6ML4B 11417108 IC50 = 82 nM T80975 C5KR0Y 11417521 IC50 = 40 nM T80975 COW7J1 11418065 IC50 = 1080 nM T80975 CH9Q2B 11418609 IC50 > 10000 nM T80975 CQD35C 11419379 IC50 = 49 nM T80975 C8TIS2 11420237 IC50 = 15 nM T80975 C73PUW 11420344 IC50 = 1 nM T80975 CO69IM 11421509 IC50 = 1 nM T80975 C5O1RM 11421633 IC50 = 3600 nM T80975 CI34BN 11428396 IC50 = 23 nM T80975 CL9J6B 11428773 IC50 = 106 nM T80975 C6LJR3 11429321 IC50 = 211 nM T80975 CREQ51 11429654 IC50 = 21 nM T80975 CY0A4E 11429729 IC50 = 18 nM T80975 CBK8Q0 11430894 IC50 = 1 nM T80975 C7AI2V 11432911 IC50 = 53 nM T80975 CYD2A6 11440253 IC50 = 110 nM T80975 C5KG7W 11440661 IC50 = 17 nM T80975 CFJ6B2 11441375 IC50 = 0.6 nM T80975 CXH8R6 11441787 IC50 = 0.5 nM T80975 C45WKC 11442803 IC50 = 22 nM T80975 C60VOM 11443129 IC50 = 2.6 nM T80975 CTCB94 11443197 IC50 = 5 nM T80975 C1LU5O 11443317 IC50 = 6 nM T80975 C2ZO1F 11443318 IC50 = 13 nM T80975 CO4F0R 11443738 IC50 > 25000 nM T80975 CT2L6G 11443940 IC50 = 7 nM T80975 C5MA4I 11444696 IC50 = 2 nM T80975 CKM8E6 11444953 IC50 = 1700 nM T80975 CAM63T 11451774 IC50 = 8 nM T80975 C8OE4T 11452154 IC50 = 6100 nM T80975 C2U9EF 11452379 IC50 = 600 nM T80975 C5E7QL 11453506 IC50 = 0.1995 nM T80975 CJC95A 11454205 IC50 > 10000 nM T80975 CL2BZ5 11454462 IC50 = 5 nM T80975 CM1CL5 11454711 Ki = 3 nM T80975 CWI62M 11454712 IC50 > 1000 nM T80975 CZ9O1A 11455031 IC50 = 29 nM T80975 CU50OG 11455909 IC50 = 5100 nM T80975 CBU5L4 11460875 Ki > 1000 nM T80975 CD97KV 11462058 IC50 = 23 nM T80975 CJUF06 11464544 IC50 = 77 nM T80975 CU0MY9 11464906 IC50 = 27 nM T80975 CJ94MR 11465254 IC50 = 390 nM T80975 C1U4GO 11465344 IC50 = 19 nM T80975 CTG3D9 11465545 IC50 = 11 nM T80975 CN20YG 11465676 IC50 = 365 nM T80975 CE5UY6 11466492 IC50 = 0.5 nM T80975 CI5KG7 11466569 IC50 = 3 nM T80975 CJ2BH4 11473904 IC50 = 67 nM T80975 C4Q7XD 11474276 IC50 = 0.8913 nM T80975 C4NR2I 11476141 IC50 = 2 nM T80975 C3J1HB 11476389 IC50 = 104 nM T80975 CU7MF2 11476903 IC50 = 35 nM T80975 CS7L5E 11477532 Ki = 2 nM T80975 C6M9NC 11477626 IC50 = 58 nM T80975 CN80LC 11477732 IC50 = 180 nM T80975 CS6GR3 11477850 IC50 = 2800 nM T80975 C85JOF 11482813 Ki = 53 nM T80975 C2Z7WP 11486459 IC50 = 1.288 nM T80975 C8XH2V 11487747 IC50 = 0.1995 nM T80975 CI59ZS 11488585 IC50 = 3.7 nM T80975 CE39WZ 11488852 IC50 = 76 nM T80975 CUC52I 11489166 Ki = 3 nM T80975 CPC9S5 11489476 IC50 = 8300 nM T80975 CS9K8W 11494006 IC50 = 430 nM T80975 C4EBN9 11494558 IC50 = 2.1 nM T80975 CXW96U 11495012 IC50 = 42 nM T80975 CK3M0T 11495270 IC50 = 2.6 nM T80975 C0H6QS 11495680 IC50 > 10000 nM T80975 CSF4Q8 11495686 IC50 = 1.3 nM T80975 C80QYI 11497471 IC50 = 2 nM T80975 C8WEO0 11502071 Ki = 8 nM T80975 CIW9L5 11502867 IC50 > 10000 nM T80975 C3ME1U 11502912 IC50 = 70 nM T80975 CD8G0U 11506240 IC50 = 7100 nM T80975 CVY9I8 11509009 IC50 = 74 nM T80975 CD6B5X 11509160 IC50 = 6.299 nM T80975 CAN05Z 11509519 IC50 = 31 nM T80975 CI0Z5J 11509810 IC50 = 110 nM T80975 CD53BX 11509997 IC50 = 1.7 nM T80975 CJP81E 11510084 IC50 = 20 nM T80975 CU2OF8 11510392 IC50 = 15 nM T80975 C29SZQ 11512193 IC50 = 20 nM T80975 CK2Q0X 11516978 IC50 > 10000 nM T80975 CRK89Q 11517130 IC50 = 206 nM T80975 CG3BZ9 11517980 IC50 = 8 nM T80975 C8AY3B 11518031 IC50 = 4 nM T80975 CLGO54 11518300 IC50 = 25 nM T80975 CA6XM4 11518397 IC50 = 110 nM T80975 CD9P5L 11518545 IC50 = 29.6 nM T80975 CIQR82 11518616 IC50 = 129 nM T80975 CMV40F 11519149 IC50 < 1 nM T80975 C87ARG 11519208 IC50 = 370 nM T80975 CX4MA8 11519486 IC50 = 11 nM T80975 C8OX7I 11523735 IC50 = 12 nM T80975 CKGD85 11526053 IC50 = 4.8 nM T80975 CO70EZ 11526166 IC50 = 800 nM T80975 CPE53F 11526238 IC50 > 10000 nM T80975 C7HMO6 11526786 IC50 > 10000 nM T80975 CN12VH 11530187 IC50 = 280 nM T80975 CL7X4Q 11530963 IC50 = 2.5 nM T80975 C5BM4T 11531799 IC50 > 10000 nM T80975 C53OSD 11532048 IC50 > 10000 nM T80975 CC4QM5 11532676 IC50 > 10000 nM T80975 CY6L8I 11532718 IC50 = 50.3 nM T80975 CI8PW4 11533783 IC50 = 16 nM T80975 C3WJZ0 11533908 IC50 = 386 nM T80975 C7T5DE 11537715 IC50 = 88 nM T80975 CWKX57 11537946 IC50 < 15 nM T80975 CTG83F 11539329 Ki > 8900 nM T80975 C8Y2BI 11540273 IC50 = 561 nM T80975 CIY5W4 11540392 IC50 = 2.4 nM T80975 C0QY6X 11540508 IC50 = 133 nM T80975 CZ68TF 11540571 IC50 = 32 nM T80975 C20ZUM 11540724 IC50 = 19 nM T80975 COS47W 11544961 IC50 = 0.6 nM T80975 CN1K3R 11545702 IC50 = 2 nM T80975 C01FVM 11546457 IC50 > 10000 nM T80975 CK48TM 11547684 IC50 = 2.6 nM T80975 CE59MD 11548497 IC50 = 26 nM T80975 CIWY62 11552514 IC50 = 3.8 nM T80975 C32PUD 11553058 IC50 = 360 nM T80975 CM72UP 11553614 IC50 = 371.9 nM T80975 CPGN98 11554757 IC50 = 5.7 nM T80975 CQV35T 11560064 IC50 = 3.8 nM T80975 CJN1E0 11561190 IC50 = 20 nM T80975 C5TJ8F 11561212 IC50 = 310 nM T80975 C3ND0O 11561658 IC50 = 2.3 nM T80975 CACS26 11561968 Ki > 4000 nM T80975 CNBM81 11562171 IC50 > 10000 nM T80975 CN49OQ 11562588 IC50 = 13.6 nM T80975 C3KWU8 11562728 IC50 = 220 nM T80975 CM7FJ1 11567496 IC50 > 1000 nM T80975 CZ1H0X 11569258 IC50 = 4600 nM T80975 CHB0U5 11569270 IC50 = 0.4 nM T80975 CJV20L 11569758 IC50 = 1.7 nM T80975 C9XI8Z 11574885 IC50 = 470 nM T80975 COGM15 11574917 IC50 > 10000 nM T80975 CGAY96 11575072 IC50 = 930 nM T80975 CP68BA 11575755 IC50 = 17 nM T80975 C2TY8V 11575947 IC50 = 184 nM T80975 CQOI76 11576375 IC50 = 9500 nM T80975 CSJ5E1 11577280 IC50 = 36 nM T80975 C5TN7O 11578019 IC50 = 4.5 nM T80975 C0HM3O 11581327 IC50 = 47 nM T80975 C8V6JD 11582722 IC50 > 1000 nM T80975 CO9KP5 11583459 IC50 = 4300 nM T80975 C4R2NM 11584238 IC50 = 5.1 nM T80975 C4PTW2 11584329 IC50 = 17 nM T80975 CR39NP 11584561 IC50 = 75.5 nM T80975 CAJQ78 11584678 IC50 = 4.7 nM T80975 CFZ1Q5 11584681 IC50 = 12 nM T80975 C3VUO7 11588815 IC50 = 1.8 nM T80975 C6DS2H 11589199 IC50 = 640 nM T80975 CZYN30 11589564 IC50 < 10 nM T80975 CA2KX0 11590078 IC50 = 5 nM T80975 C6FG3R 11590287 IC50 = 101.2 nM T80975 CMIL86 11590363 Ki > 8900 nM T80975 CB08WI 11590515 IC50 = 4 nM T80975 CWAZ43 11591353 IC50 = 17 nM T80975 CONZ37 11591872 IC50 = 7 nM T80975 C1YIG3 11592064 IC50 = 18.6 nM T80975 C2N4XP 11595595 IC50 = 30 nM T80975 C0NV9Y 11596881 IC50 > 10000 nM T80975 C9Z1SG 11597872 IC50 = 53.5 nM T80975 CNE0J2 11598750 IC50 = 13.7 nM T80975 C6C9WI 11598848 IC50 = 17 nM T80975 CFPB69 11599241 IC50 = 289 nM T80975 CW0RG9 11599334 IC50 = 15.3 nM T80975 C34PKN 11602733 IC50 = 12.7 nM T80975 C45BMY 11603130 IC50 = 4200 nM T80975 CFN80A 11603296 IC50 = 1.5 nM T80975 C7I3CP 11603633 IC50 = 5.1 nM T80975 C1TP3Q 11603793 IC50 = 150 nM T80975 C69FYK 11604142 Ki = 85 nM T80975 C0N5DY 11604763 IC50 = 66 nM T80975 CM0RQ8 11605387 IC50 = 52.4 nM T80975 C6ZRQ0 11605787 IC50 = 6.4 nM T80975 CKW49P 11605989 IC50 = 6300 nM T80975 CU2NX1 11606286 IC50 = 3.6 nM T80975 CA3MB5 11610147 IC50 = 2.2 nM T80975 CDV1B5 11610420 IC50 = 12 nM T80975 CLWA52 11611374 IC50 = 73 nM T80975 CWPR69 11612103 IC50 = 24.8 nM T80975 C1SL7N 11612461 IC50 = 20 nM T80975 CU6T2L 11613133 IC50 = 160 nM T80975 CL5OY4 11613524 IC50 = 10 nM T80975 CPTE09 11616279 IC50 = 8200 nM T80975 CV71YX 11617549 IC50 = 110 nM T80975 CY6SW0 11617856 IC50 = 435 nM T80975 C1BLZ5 11620055 IC50 > 10000 nM T80975 CUO43M 11620207 IC50 = 390 nM T80975 C5B3XJ 11620410 Ki = 2.8 nM T80975 CG1JN5 11620467 IC50 = 210 nM T80975 CCYV36 11620477 IC50 = 300 nM T80975 CI1FZ4 11624999 IC50 = 1.1 nM T80975 CVQ42G 11625281 IC50 = 4.4 nM T80975 CHJ1W9 11625507 IC50 = 30.1 nM T80975 CGU3P6 11625750 IC50 = 7.1 nM T80975 C70LDZ 11625929 IC50 < 1 nM T80975 C9ZD2E 11626406 IC50 = 537 nM T80975 CSM62L 11626920 IC50 > 30000 nM T80975 CJ1DK9 11627158 IC50 = 150 nM T80975 CWM80X 11627419 IC50 = 1100 nM T80975 C6CEX2 11627663 IC50 = 5.8 nM T80975 C9UF2Y 11627875 IC50 = 298.6 nM T80975 CR67IJ 11628038 IC50 = 1.5 nM T80975 CK34LS 11632737 IC50 = 40 nM T80975 C51EYB 11634026 IC50 = 4.8 nM T80975 CX80WU 11634758 IC50 = 6.9 nM T80975 C1TZY3 11635079 IC50 = 57 nM T80975 C4QKF9 11639559 IC50 = 29 nM T80975 CFM2Y4 11640405 IC50 = 1000 nM T80975 C9T6SC 11640926 Ki > 8900 nM T80975 CVH29N 11642023 IC50 = 890 nM T80975 C4GTZ8 11645322 IC50 = 350 nM T80975 C74MPT 11646161 IC50 = 1 nM T80975 CEVM71 11647279 IC50 = 481 nM T80975 CTNK57 11648060 IC50 = 177 nM T80975 C9FJM8 11648430 IC50 = 133 nM T80975 C0RNY2 11653701 IC50 = 18 nM T80975 CU1PC4 11653702 IC50 = 20 nM T80975 CZF82K 11653746 IC50 = 1.2 nM T80975 CNC75B 11653889 IC50 = 240.9 nM T80975 CJRA63 11654668 IC50 < 1 nM T80975 C9SPF4 11654839 IC50 > 10000 nM T80975 C63JRY 11655241 IC50 > 10000 nM T80975 CG2O8J 11655538 IC50 = 16 nM T80975 CRV5D2 11655925 IC50 = 58 nM T80975 CHRP74 11656019 IC50 = 3.4 nM T80975 C3L2HT 11656560 IC50 = 1700 nM T80975 CX7C1T 11656606 IC50 = 100 nM T80975 CU1I9G 11656638 IC50 = 57.4 nM T80975 CK9Q3G 11660444 IC50 = 2.9 nM T80975 CB4J1E 11660744 IC50 = 1.1 nM T80975 C1AUX0 11661290 IC50 = 1300 nM T80975 C3H7JL 11661794 IC50 = 13.5 nM T80975 CG54AP 11661821 IC50 = 24 nM T80975 C24GRQ 11661959 IC50 > 10000 nM T80975 C0PM8X 11662019 IC50 = 64 nM T80975 C7QI5P 11662096 IC50 = 5 nM T80975 CI8V3C 11662097 IC50 = 3 nM T80975 CQ47BI 11662314 IC50 = 290 nM T80975 CWJR63 11662632 IC50 = 110.5 nM T80975 C0DCW6 11662695 IC50 = 0.9 nM T80975 CPB09V 11663290 IC50 = 160 nM T80975 C8RMT2 11663885 IC50 = 67 nM T80975 C43JZK 11668206 IC50 = 1890 nM T80975 C4C3UB 11668255 IC50 = 17 nM T80975 CP92IG 11668816 IC50 = 28.7 nM T80975 CCGO58 11669282 IC50 = 169 nM T80975 C7ZG5I 11670166 IC50 = 23.6 nM T80975 COR60S 11670781 IC50 = 2.2 nM T80975 CPME86 11670863 IC50 = 13 nM T80975 CALI63 11671030 IC50 = 9 nM T80975 CVLA25 11675714 IC50 > 10000 nM T80975 CX04MA 11676364 IC50 = 14 nM T80975 C9L0KU 11676434 IC50 = 4.5 nM T80975 CC8SJ3 11676616 IC50 = 590 nM T80975 CB58TO 11676719 IC50 = 1.9 nM T80975 CFG17W 11677639 IC50 > 1000 nM T80975 CW9B8E 11678175 IC50 > 25000 nM T80975 CX5N6F 11681911 IC50 = 6 nM T80975 CCX2F5 11682611 IC50 = 14 nM T80975 CS72ED 11682843 IC50 > 10000 nM T80975 CU6T4Z 11683186 IC50 = 111.9 nM T80975 CEOD83 11683384 IC50 = 236.5 nM T80975 C5FI8Q 11683484 IC50 < 1 nM T80975 CPS06C 11683901 IC50 = 10.3 nM T80975 CP3U0W 11684933 IC50 = 3096 nM T80975 CYO6X9 11684994 Ki = 380 nM T80975 C8AEX7 11687971 IC50 = 30300 nM T80975 CCEY64 11689855 IC50 = 6 nM T80975 CU0E8O 11690457 Ki > 4000 nM T80975 C7I9FP 11690513 IC50 > 10000 nM T80975 C2L9JU 11690518 IC50 = 2.4 nM T80975 CLC53E 11691173 IC50 > 10000 nM T80975 CP8WJ3 11691483 IC50 = 31.2 nM T80975 CI3EO4 11692100 IC50 = 4700 nM T80975 CXL42T 11696630 IC50 = 14 nM T80975 C15XRO 11697767 IC50 = 15.8 nM T80975 CPJ94X 11698403 IC50 = 67.1 nM T80975 CU6D3X 11703421 IC50 = 20 nM T80975 CFTN64 11704732 IC50 = 9 nM T80975 CB0AP2 11705863 Ki > 4000 nM T80975 CJ8ZI5 11710567 IC50 = 1 nM T80975 C6WMG4 11710853 IC50 = 3 nM T80975 C7HJO5 11710909 IC50 = 1.5 nM T80975 CW8L4M 11711658 IC50 = 2 nM T80975 C0WKF6 11711734 IC50 = 17 nM T80975 CHL5W3 11712625 IC50 = 2.2 nM T80975 C9ROB0 11713267 IC50 = 11 nM T80975 C0OWS4 11713310 IC50 = 10 nM T80975 CN5UX7 11713409 IC50 = 14 nM T80975 C5A3BH 11717763 IC50 = 0.7 nM T80975 C1FTX3 11719305 IC50 > 10000 nM T80975 CZY05V 11719421 IC50 = 555 nM T80975 C9R0FW 11719590 IC50 = 30 nM T80975 C8BX7M 11720813 IC50 = 230 nM T80975 CRZ4K6 11724734 IC50 > 100000 nM T80975 CP1WX2 11725783 IC50 = 26 nM T80975 C9P0VD 11729539 IC50 > 100000 nM T80975 CY89WV 11736130 Ki > 1000 nM T80975 C01GBO 11738453 IC50 > 10000 nM T80975 CU5V9K 11749082 IC50 = 3 nM T80975 CS5QL4 11749561 IC50 = 3.8 nM T80975 CV64JS 11750694 IC50 = 0.37 nM T80975 C8MOK3 11750699 IC50 < 1000 nM T80975 C67ERD 11752517 Ki = 4 nM T80975 CS9WP2 11752657 IC50 = 15000 nM T80975 CN8S1E 11752715 IC50 = 6600 nM T80975 CTRV89 11753309 Ki = 0.5 nM T80975 CE0KI4 11753519 IC50 = 18500 nM T80975 CP7AH3 11755812 IC50 = 33 nM T80975 C7C6BM 11772612 IC50 = 3 nM T80975 CM86DJ 11775224 IC50 = 40 nM T80975 C2GCB7 11779327 IC50 = 7600 nM T80975 CL87KR 11785748 IC50 = 1900 nM T80975 C4NO7Y 11809063 IC50 = 414 nM T80975 C4Q1AE 11817879 IC50 > 10000 nM T80975 CCI6R5 11842847 IC50 = 4800 nM T80975 CMO6N4 11842849 IC50 = 590 nM T80975 C9HT7B 11842850 IC50 = 1900 nM T80975 CP6KY2 11843009 IC50 = 170 nM T80975 C8FHK9 11843010 IC50 = 220 nM T80975 C7D6MQ 11843012 IC50 = 170 nM T80975 C4T2WC 11843013 IC50 = 210 nM T80975 CS36BH 11843159 IC50 = 140 nM T80975 C7DU6T 11843160 IC50 = 620 nM T80975 CH6W3V 11844349 IC50 = 190 nM T80975 CI15NA 11844350 IC50 = 420 nM T80975 CUL2C8 11844485 IC50 = 130 nM T80975 C96ORQ 11844486 IC50 = 140 nM T80975 C4SK3L 11844487 IC50 = 260 nM T80975 C6KF8Z 11844488 IC50 = 230 nM T80975 C9ECK3 11844489 IC50 = 230 nM T80975 C83YRX 11844616 IC50 = 590 nM T80975 CV24WL 11844764 IC50 = 190 nM T80975 C9JT4S 11847343 IC50 = 162 nM T80975 CAZS08 11848309 IC50 = 1145 nM T80975 C43IVN 11848567 IC50 = 6292 nM T80975 C9LAY8 11848825 IC50 = 8553 nM T80975 CN1U7P 11855937 IC50 = 23 nM T80975 CYA0X2 11856199 IC50 = 19 nM T80975 C0A9WL 11856200 IC50 = 806 nM T80975 CJ5G9Y 11856201 IC50 = 8 nM T80975 COLP81 11856204 IC50 = 15 nM T80975 CSRQ05 11856467 IC50 = 71 nM T80975 CA2BL5 11856735 IC50 = 179 nM T80975 CI7DT1 11857432 Ki > 1300 nM T80975 CBT94Q 11857507 Ki = 56 nM T80975 CEA7I9 11857949 Ki = 382 nM T80975 CHR92S 11858109 Ki = 139 nM T80975 CDKH57 11858286 Ki > 3000 nM T80975 C8NF6H 11947782 Ki = 2020 nM T80975 CC09DE 11955790 IC50 = 140 nM T80975 C2YDO7 11957783 IC50 = 951 nM T80975 CO8QR4 11962890 Ki = 1980 nM T80975 C0HE1D 11962891 Ki = 35.9 nM T80975 CFP7M5 11962976 Ki = 932 nM T80975 CP89KY 11962977 Ki = 382 nM T80975 CCY4J2 11962978 Ki = 38 nM T80975 C3XWU1 11963015 Ki = 452 nM T80975 CA7Y5P 11963057 Ki = 234 nM T80975 CTC31Z 11963059 IC50 = 143 nM T80975 C3H4PA 11963103 Ki = 74.1 nM T80975 CI7G5W 11963258 Ki = 541 nM T80975 CT1RA7 11963259 Ki = 1240 nM T80975 CY8GD6 11963300 Ki = 1310 nM T80975 CQ2WD1 11963302 Ki = 903 nM T80975 CGCX39 11963344 Ki > 6600 nM T80975 C4O3UR 11963386 Ki = 1380 nM T80975 CPG89E 11963387 Ki = 945 nM T80975 CF3W2N 11963388 Ki = 2720 nM T80975 CQT2I1 11963389 Ki = 588 nM T80975 CT91NG 11963423 Ki = 501 nM T80975 CH2A1C 11963425 Ki = 4730 nM T80975 CSC8A9 11973903 IC50 > 5000 nM T80975 CB60GC 11974016 IC50 = 5500 nM T80975 CZG6O4 11974017 IC50 = 100 nM T80975 CUBL61 11974019 IC50 = 2500 nM T80975 C15HWQ 11974020 IC50 = 500 nM T80975 CYLH02 11974021 IC50 = 650 nM T80975 C2RSN3 11974115 IC50 = 50 nM T80975 CY37WX 11974116 IC50 = 5000 nM T80975 CXQ7Y1 11974120 IC50 > 20000 nM T80975 C3Z1JF 11974212 IC50 > 10000 nM T80975 C5OX6U 11974213 IC50 = 1200 nM T80975 CF2P7Z 11974214 IC50 = 10000 nM T80975 C0GZL5 11974215 IC50 = 6500 nM T80975 CDZ1I3 11989153 IC50 = 405.5 nM T80975 CY4R6F 11990802 IC50 = 2.7 nM T80975 CM50UH 12000646 IC50 = 147 nM T80975 CJ5K4M 12341776 IC50 = 4.5 nM T80975 CU4C3V 12968172 IC50 = 16900 nM T80975 CI8VE5 12968173 IC50 = 1600 nM T80975 CR75GZ 12968174 IC50 = 3350 nM T80975 CEVY69 12968175 IC50 = 3200 nM T80975 CL1PR6 12968176 IC50 = 1080 nM T80975 CY5EA7 12968177 IC50 = 1860 nM T80975 CZ98FV 12968178 IC50 = 4240 nM T80975 C4SUK6 12968179 IC50 = 677 nM T80975 CGIZ84 12968180 IC50 = 9820 nM T80975 C5MX8N 12968181 IC50 = 9110 nM T80975 C5MI4N 14246200 IC50 = 1560 nM T80975 C2Z8DQ 14624081 IC50 > 10000 nM T80975 CDGF78 15282555 IC50 = 1200 nM T80975 CP8OW6 15858662 IC50 > 1000 nM T80975 C24FXN 15941243 IC50 = 888 nM T80975 CG5IO2 15941244 IC50 = 126 nM T80975 C8Y1XP 15941246 IC50 = 3 nM T80975 CB94LR 15941247 IC50 = 65 nM T80975 CZ38JG 15941390 IC50 = 6 nM T80975 CE57UJ 15941392 IC50 = 4 nM T80975 C1AIM6 15941393 IC50 = 6 nM T80975 CN7PO9 15941394 IC50 = 19 nM T80975 C9E3RP 15941395 IC50 = 5 nM T80975 CSBF70 15941529 IC50 = 110 nM T80975 CQM93O 15941530 IC50 = 49 nM T80975 C0M7TW 15948947 IC50 = 20 nM T80975 C1VNB4 15948949 IC50 = 66 nM T80975 CH8ZG5 15949048 IC50 = 5 nM T80975 C35LRO 15949471 IC50 = 51 nM T80975 CK2Z6Y 15949521 IC50 = 280 nM T80975 CBZF29 15949522 IC50 = 576 nM T80975 C34MCY 15949523 IC50 = 43 nM T80975 CS3P9G 15949524 IC50 = 30 nM T80975 C1KPH2 15949525 IC50 = 9069 nM T80975 CV4EZ6 15949611 IC50 = 3.7 nM T80975 C7LB4I 15949613 Ki = 0.024 nM T80975 C5JG9R 15949617 IC50 = 4 nM T80975 C8FT6U 15949618 IC50 = 451 nM T80975 C30PVQ 15949619 IC50 = 48 nM T80975 C3PNO2 15949620 IC50 = 63 nM T80975 C4I5RS 15949621 IC50 > 10000 nM T80975 CVJ9A0 15949712 IC50 = 356 nM T80975 CEI2K8 15949887 IC50 = 1012 nM T80975 CAIN63 15949888 IC50 > 10000 nM T80975 C2VDI1 15949889 IC50 = 590 nM T80975 COC02T 15949890 IC50 = 1712 nM T80975 CFQ6X3 15949974 IC50 = 605 nM T80975 CMKZ23 15949975 IC50 = 1726 nM T80975 CWM5L4 15949976 IC50 = 582 nM T80975 CO7NG2 15950141 IC50 = 885 nM T80975 COIG45 15950224 IC50 = 36 nM T80975 C9V0TO 15950311 IC50 = 55 nM T80975 C9RQN8 15950748 IC50 = 125 nM T80975 CSK90Y 15991573 IC50 = 2 nM T80975 CPNW35 15991575 IC50 = 306 nM T80975 C12WCK 16004702 IC50 = 1.7 nM T80975 CFPW41 16007116 Ki > 8900 nM T80975 C8PRQ6 16040281 IC50 = 61 nM T80975 CFWR47 16040288 IC50 >= 5000 nM T80975 C7NCA6 16040289 Ki = 10 nM T80975 C4MQU1 16040290 IC50 = 310 nM T80975 CU0S5T 16040363 IC50 = 12 nM T80975 CK4LA5 16040525 IC50 = 7 nM T80975 C5K3RO 16040526 IC50 = 3 nM T80975 C9C3AE 16040527 IC50 = 14 nM T80975 CYXZ47 16040697 IC50 = 14 nM T80975 CC68WU 16040698 IC50 = 3 nM T80975 CI0U9N 16040699 IC50 = 31 nM T80975 CYT5V7 16040870 IC50 = 6 nM T80975 CTG84Q 16041065 IC50 = 57 nM T80975 C93MID 16041066 IC50 = 6 nM T80975 CX1SD5 16041234 IC50 = 10 nM T80975 CWC7B6 16041238 IC50 = 170 nM T80975 CE9ZW5 16041961 IC50 = 7 nM T80975 CD85IU 16041962 IC50 = 18 nM T80975 CEDC74 16042706 IC50 = 9 nM T80975 CMB30J 16042707 IC50 = 1 nM T80975 C8NME0 16042894 IC50 = 15 nM T80975 CQR5O7 16042971 IC50 = 6300 nM T80975 CZI2H3 16043068 IC50 = 13 nM T80975 CQI0A5 16043229 IC50 = 11 nM T80975 CZKD04 16043241 IC50 = 1 nM T80975 C9X4TQ 16043242 IC50 = 8 nM T80975 CD2F8V 16046116 IC50 > 10000 nM T80975 C9TU1O 16046126 IC50 > 1000 nM T80975 CI74HE 16049888 IC50 = 5 nM T80975 CW2XK6 16050925 IC50 = 800 nM T80975 CRM8E0 16066844 IC50 = 42 nM T80975 CKV4G1 16079040 IC50 = 660 nM T80975 C3ZV2X 16086076 IC50 = 173 nM T80975 C0SO7D 16086077 IC50 = 103 nM T80975 C0WU9I 16086078 IC50 = 6 nM T80975 CVE6C8 16086088 IC50 = 1 nM T80975 CH1R8K 16086091 IC50 = 5 nM T80975 CT4RS8 16086092 IC50 = 52 nM T80975 CZ2QU1 16086093 IC50 = 1438 nM T80975 C13OVU 16086099 IC50 = 8 nM T80975 C2YC0S 16086100 IC50 = 48 nM T80975 C28UZX 16086101 IC50 = 8 nM T80975 CKM8E4 16086102 IC50 = 3 nM T80975 CF0N4J 16086103 IC50 = 21 nM T80975 CKR57M 16086104 IC50 = 17 nM T80975 CI5HJ8 16086105 IC50 = 1415 nM T80975 C68SBO 16086106 IC50 = 461 nM T80975 CAYV39 16086107 IC50 = 47 nM T80975 C06NOI 16086108 IC50 = 360 nM T80975 C16NRY 16086114 IC50 = 1 nM T80975 C87TPW 16086115 IC50 = 15 nM T80975 CW35LJ 16086116 IC50 = 7 nM T80975 CA3BD7 16086117 IC50 = 292 nM T80975 C3EKF4 16086118 IC50 = 246 nM T80975 C0QCG4 16086142 IC50 = 4 nM T80975 C20DST 16105503 IC50 > 300 nM T80975 CCN62F 16105510 IC50 > 300 nM T80975 C73MLJ 16108977 IC50 = 3 nM T80975 C01GIO 16108981 IC50 > 25000 nM T80975 C6FO0H 16108986 IC50 = 59 nM T80975 CXI9C8 16108987 IC50 = 705 nM T80975 CEC7P3 16108988 IC50 = 100 nM T80975 CGK5O8 16108989 IC50 = 1300 nM T80975 C5SE6X 16108990 IC50 > 25000 nM T80975 C03GLR 16108991 IC50 = 70 nM T80975 C3L6TH 16108992 IC50 > 25000 nM T80975 COEI61 16108993 IC50 > 25000 nM T80975 C39YWL 16108994 IC50 > 25000 nM T80975 C9IX0U 16108995 IC50 = 461 nM T80975 CU2TK3 16108996 IC50 > 25000 nM T80975 CA2U9H 16108997 IC50 = 46 nM T80975 CX21ZN 16108999 IC50 = 4000 nM T80975 CF57NZ 16109000 IC50 > 25000 nM T80975 CQG45C 16109001 IC50 = 7800 nM T80975 C3L8KE 16109002 IC50 > 8000 nM T80975 CM40ZW 16109003 IC50 > 25000 nM T80975 C8P4ZK 16109016 IC50 < 1 nM T80975 CY1E3Q 16109017 IC50 > 1000 nM T80975 CV7S6Z 16109018 IC50 = 480 nM T80975 CB98HV 16109019 IC50 = 810 nM T80975 C49VTS 16109020 IC50 = 1010 nM T80975 C6FZ7A 16109023 IC50 = 1 nM T80975 CWS8D0 16109024 IC50 = 4 nM T80975 C1WS6E 16109034 IC50 > 1000 nM T80975 C8IES6 16109035 IC50 = 170 nM T80975 C1U8XW 16109036 IC50 = 1030 nM T80975 CNG5L6 16109037 IC50 = 3000 nM T80975 C34KRB 16109040 IC50 = 1 nM T80975 CZ5Y3V 16116847 IC50 = 947 nM T80975 CLO43V 16116849 IC50 > 5000 nM T80975 C0HO6T 16118191 IC50 = 41 nM T80975 CT92BZ 16118192 IC50 = 120 nM T80975 CIZ6B4 16118193 IC50 = 17 nM T80975 C2CN5O 16118323 IC50 = 32 nM T80975 C4GTU3 16118324 IC50 = 272 nM T80975 CXC78K 16118603 IC50 = 587 nM T80975 CI4E6Y 16118605 IC50 > 8300 nM T80975 C8LIW4 16118609 IC50 > 8300 nM T80975 CGC34R 16118737 IC50 = 24 nM T80975 CAN2K6 16118739 IC50 > 25000 nM T80975 C1VQ0J 16124774 IC50 = 87 nM T80975 CX7FV0 16124775 IC50 = 55 nM T80975 CGF2M4 16124831 IC50 = 36 nM T80975 CU1K9R 16124836 IC50 = 1300 nM T80975 C3FS0I 16124974 IC50 = 12 nM T80975 C3B8SQ 16124975 IC50 = 31 nM T80975 CD3U0I 16124976 IC50 = 15 nM T80975 CTY7Z5 16125041 IC50 = 3200 nM T80975 CDEZ21 16125042 IC50 = 18 nM T80975 C5W9ZT 16125110 IC50 = 4620 nM T80975 C9R4EN 16125232 IC50 = 12 nM T80975 C9XMJ4 16125233 IC50 = 4 nM T80975 C4BFJ3 16125303 IC50 = 3090 nM T80975 CF23VU 16125380 IC50 = 3 nM T80975 CZM0J2 16125381 IC50 = 26 nM T80975 CVAZ06 16125453 IC50 = 35 nM T80975 CLV30K 16125513 IC50 = 12000 nM T80975 C3E5OB 16125514 IC50 = 465 nM T80975 C5VPH9 16129448 IC50 = 886 nM T80975 CZ08YH 16214904 IC50 = 760 nM T80975 CK8Z9L 16220221 IC50 = 38 nM T80975 CFI8G2 16220223 IC50 = 10 nM T80975 CTU7J0 16220225 IC50 = 7960 nM T80975 C7SE5O 16220227 IC50 > 50000 nM T80975 C9GU5M 16220228 IC50 = 108 nM T80975 C27GFI 16220230 IC50 = 962 nM T80975 CCW65G 16220231 IC50 = 197 nM T80975 CN6G4O 16220232 IC50 = 22 nM T80975 C0ZUH7 16220280 IC50 = 75 nM T80975 C39SIQ 16220281 IC50 = 8 nM T80975 CP3HS4 16220354 IC50 = 6 nM T80975 CJ2PR1 16220790 IC50 = 2370 nM T80975 C0JA4Q 16220791 IC50 = 8 nM T80975 CWIT69 16220793 IC50 = 85 nM T80975 CI84RL 16220795 IC50 = 101 nM T80975 C3W1LK 16220874 IC50 = 36 nM T80975 CUNW89 16220876 IC50 = 78 nM T80975 C1VUC5 16220877 IC50 = 33 nM T80975 CN91VO 16220879 IC50 = 54 nM T80975 CVQ9T5 16220880 IC50 = 48 nM T80975 C1U9XM 16220882 IC50 = 28 nM T80975 CZUQ73 16220957 IC50 = 3 nM T80975 CA5NX6 16220959 IC50 = 10 nM T80975 C8J3YN 16220960 IC50 = 5 nM T80975 CPV4G2 16220962 IC50 = 69 nM T80975 C4L7QD 16221024 IC50 = 11 nM T80975 CAU7E0 16221025 IC50 = 18 nM T80975 C4GPA2 16221027 IC50 = 29 nM T80975 C3SH0K 16221088 IC50 = 40 nM T80975 CM8N1R 16221090 IC50 = 10 nM T80975 C5E6AC 16221091 IC50 = 195 nM T80975 CXL6V8 16221092 IC50 = 20 nM T80975 CW35VX 16221140 IC50 = 15 nM T80975 C78VJQ 16221258 IC50 = 45 nM T80975 C9X2GY 16221259 IC50 = 11 nM T80975 CBH1I9 16221317 IC50 = 50 nM T80975 C3P7XC 16221373 IC50 = 4680 nM T80975 CJ8RC1 16221375 IC50 = 2 nM T80975 C5TV3A 16221425 IC50 = 10 nM T80975 C8CKV2 16221426 IC50 = 124 nM T80975 CQE9N1 16221427 IC50 = 2140 nM T80975 CU56EW 16664858 IC50 > 10000 nM T80975 CAK1C4 16666757 IC50 > 100000 nM T80975 C1QRG8 16666806 IC50 = 11260 nM T80975 CF8B5S 16666857 IC50 = 1100 nM T80975 C5U8LG 16666858 IC50 = 142 nM T80975 CJ9C7N 16666859 IC50 = 56 nM T80975 C5JQ6H 16666860 IC50 = 65 nM T80975 C4VW0O 16666861 IC50 = 74 nM T80975 C1IO4K 16666862 IC50 = 144 nM T80975 CS1LR2 16666908 IC50 = 30 nM T80975 CI32LX 16666909 IC50 = 119 nM T80975 C07BIL 16666910 IC50 = 1100 nM T80975 C71TSX 16666911 IC50 = 14 nM T80975 C2IF3P 16678352 IC50 = 4210 nM T80975 C3IO1C 16679060 IC50 > 10000 nM T80975 CPZ65H 16717966 IC50 = 11 nM T80975 CY1E2N 16723801 IC50 = 26000 nM T80975 C0VUQ3 16727122 IC50 = 16 nM T80975 C0V8FB 16730091 IC50 = 4718 nM T80975 CA24TE 16730092 IC50 = 2481 nM T80975 C9IW5S 16730105 IC50 = 73 nM T80975 C0H8UN 16730109 IC50 > 10000 nM T80975 C6S3YO 16731782 IC50 = 69 nM T80975 CK9CV4 16733534 IC50 > 5000 nM T80975 CP1RF4 16739311 IC50 = 16 nM T80975 C72THB 16739368 IC50 > 100000 nM T80975 C1Y2JH 16745310 IC50 = 378.7 nM T80975 CZY73G 16747388 EC50 = 4200 nM T80975 CDZ31W 16747696 IC50 = 10 nM T80975 CU5Q9B 16757524 IC50 = 921 nM T80975 C9BJ7Q 16757577 IC50 = 91000 nM T80975 C75HUG 16759369 IC50 = 2 nM T80975 CV7Q2B 16876702 IC50 = 5200 nM T80975 CL9BQ6 17748275 IC50 = 1002 nM T80975 C4YL0X 17755115 Ki = 48 nM T80975 C8FP3L 17755116 Ki = 3.9 nM T80975 C0X7FU 17755117 Ki = 2 nM T80975 CI10AY 17755137 IC50 = 32 nM T80975 CNJV57 17755212 Ki = 9 nM T80975 CJ7A9U 17755213 Ki = 287 nM T80975 CTGO63 17755214 Ki = 17 nM T80975 CTR83O 17755215 Ki = 40 nM T80975 CLB1D9 17755216 Ki = 128 nM T80975 C4HLX0 17755232 IC50 = 42 nM T80975 CU9MH8 17755233 IC50 = 33 nM T80975 C8M6LZ 17755310 Ki = 12 nM T80975 C6H4QO 17755311 Ki = 4 nM T80975 CIB08M 17755312 Ki = 0.5 nM T80975 C3NR5D 17755313 Ki = 0.5 nM T80975 C75UXW 17755314 Ki = 3.6 nM T80975 CIS52L 17755330 IC50 = 230 nM T80975 C5PU1S 17755399 Ki = 25 nM T80975 CR0K4I 17755400 Ki = 20 nM T80975 CQ5D9H 17755420 IC50 = 4.8 nM T80975 CQ19GV 17755641 IC50 = 190 nM T80975 CL39DG 17755642 IC50 = 105 nM T80975 CK61TQ 17755722 Ki = 160 nM T80975 CA6FO3 17755723 Ki = 1 nM T80975 C01YSP 17755724 Ki = 3 nM T80975 C1JFM0 17755746 IC50 = 16 nM T80975 C1L5IA 17755861 IC50 = 1.5 nM T80975 C28TDB 17756743 IC50 = 2600 nM T80975 CV1DQ3 18070506 IC50 = 84.9 nM T80975 C4YL8A 18205340 IC50 = 980 nM T80975 CZB5L4 18382784 IC50 = 140 nM T80975 C6JGI7 18450541 IC50 = 22 nM T80975 CLF1D3 18450549 IC50 = 94 nM T80975 CN0SA1 18450585 IC50 = 6 nM T80975 C4D6VY 18450694 IC50 = 11 nM T80975 C7H4UM 18450846 IC50 = 1 nM T80975 C0KJM1 18450928 IC50 = 250 nM T80975 CV3A0P 18450940 IC50 = 27 nM T80975 CJA0D6 18451024 IC50 > 50000 nM T80975 C6FQB7 18451036 IC50 > 50000 nM T80975 CB9LG5 18451073 IC50 = 2 nM T80975 CSJ97R 18451176 IC50 = 7 nM T80975 CC9HG2 18451200 IC50 = 8 nM T80975 CQ1F3W 18451228 IC50 = 9 nM T80975 CP5EF3 18451249 IC50 = 11 nM T80975 CL89ZM 18451253 IC50 = 388 nM T80975 CW05LC 18451306 IC50 = 13 nM T80975 CY89DE 18451351 IC50 = 520 nM T80975 C6JLN5 18451354 IC50 = 12000 nM T80975 CV8K0J 18451356 IC50 = 75 nM T80975 C71YIX 18451361 IC50 = 152 nM T80975 CQL17F 18451362 IC50 = 15 nM T80975 CQTB81 18451364 IC50 = 41 nM T80975 C2CB7I 18451365 IC50 = 16 nM T80975 COY36H 18451370 IC50 = 45 nM T80975 C5WXF6 18451372 IC50 = 147 nM T80975 CO8IU6 18451373 IC50 = 410 nM T80975 CMQD24 18451374 IC50 = 9 nM T80975 C3RB2Y 18451383 IC50 = 26 nM T80975 CF01AU 18451385 IC50 = 491 nM T80975 CX4TA1 18451386 IC50 = 420 nM T80975 CIZE32 18451387 IC50 = 4900 nM T80975 C5J8AQ 18451388 IC50 = 23 nM T80975 CY01DL 18451389 IC50 = 56 nM T80975 CIJ75W 18451390 IC50 = 30 nM T80975 C3SJ0Y 18451391 IC50 = 38 nM T80975 CZ90RF 18516895 IC50 = 82 nM T80975 CHVU30 18516919 IC50 = 200 nM T80975 CQO3F4 18516938 IC50 = 94 nM T80975 CFAY17 18516981 IC50 = 55 nM T80975 CJZR02 18567634 IC50 = 4.2 nM T80975 CGZ49R 18732328 IC50 > 12500 nM T80975 CSK5L4 18770844 IC50 > 10000 nM T80975 C5WAV7 19597382 IC50 = 500 nM T80975 CU5CK6 19597400 IC50 = 7100 nM T80975 CZQ92B 19597433 IC50 = 430 nM T80975 C02JLX 19597448 IC50 = 900 nM T80975 CYIX85 19597450 IC50 = 90 nM T80975 CFH4I2 19597457 IC50 = 900 nM T80975 C0JQ7H 19597465 IC50 = 1310 nM T80975 CP01WN 19597468 IC50 = 1000 nM T80975 CA09JB 19597476 IC50 = 3300 nM T80975 CC78WA 19597518 IC50 > 50000 nM T80975 CV0U1N 19597532 IC50 = 400 nM T80975 C1B3DX 19597536 IC50 = 2000 nM T80975 CJX9G0 20773396 Ki = 9 nM T80975 CTL37J 20773471 Ki = 259 nM T80975 C2NT0H 20773474 Ki = 23 nM T80975 CH4K5Y 20824932 IC50 = 17 nM T80975 CQ91KY 21049437 IC50 = 21 nM T80975 C3FA9D 21059967 IC50 = 41 nM T80975 C6RQ2N 21060773 IC50 = 107 nM T80975 CH4B5K 21081523 IC50 > 5000 nM T80975 C25UKC 21081761 IC50 = 4.27 nM T80975 CL81VC 21100709 IC50 = 5960 nM T80975 CJL83T 21260277 IC50 = 150 nM T80975 C60QKI 21260292 IC50 = 210 nM T80975 CUH32C 21260305 IC50 = 9.5 nM T80975 CA51HY 21701560 IC50 = 58 nM T80975 CVI49J 21701562 IC50 = 460 nM T80975 C3VT6O 21701572 IC50 = 20 nM T80975 CFN6G4 21701597 IC50 = 20 nM T80975 C3A8EN 21934593 IC50 = 15 nM T80975 CMSV01 21934607 IC50 = 10 nM T80975 CKN5J1 21934616 IC50 = 10 nM T80975 CB41RG 21934630 IC50 = 34 nM T80975 C49ZWS 21934637 IC50 = 13 nM T80975 C8M3CQ 21934651 IC50 = 27 nM T80975 CIS25P 21934657 IC50 = 10 nM T80975 C42UZF 21934662 IC50 = 9 nM T80975 CFRH31 21934687 IC50 = 557 nM T80975 CCZO61 21934688 IC50 = 153 nM T80975 C8DWX1 21934697 IC50 = 9 nM T80975 CG60BL 21934707 IC50 = 16 nM T80975 C5JZX0 21945905 IC50 = 90 nM T80975 CME79P 21945942 IC50 = 150 nM T80975 C76PDN 21945971 IC50 = 52 nM T80975 CK8X7S 21956341 IC50 = 0.6 nM T80975 CB87EW 21957795 IC50 = 31000 nM T80975 C7ST6F 22019143 IC50 = 85 nM T80975 CC67ZF 22059355 IC50 = 37 nM T80975 CPV5Z0 22132688 IC50 = 40 nM T80975 CDS7B0 22172654 IC50 > 10000 nM T80975 C6G4JM 22172657 IC50 = 2300 nM T80975 CFHP82 22249429 Ki = 4 nM T80975 C6GX1O 22249432 Ki = 8 nM T80975 CXI15H 22249458 Ki > 20000 nM T80975 CXT75P 22249467 Ki = 2 nM T80975 CV4IR1 22260308 IC50 = 40 nM T80975 CLJN24 22260328 IC50 = 30 nM T80975 CA2C0U 22273608 IC50 = 30 nM T80975 CG18XD 22273633 IC50 = 13 nM T80975 CF6LA9 22478260 IC50 = 8 nM T80975 CMRO51 22478297 IC50 = 40 nM T80975 C8JP9Y 22605351 IC50 = 9 nM T80975 CY0G8V 22624897 IC50 < 2 nM T80975 C2P1DL 22667101 IC50 = 90 nM T80975 CK35BP 22667145 IC50 = 400 nM T80975 CSB1G3 22692751 IC50 = 1170 nM T80975 CYN49O 22692759 IC50 = 1990 nM T80975 CZRM03 22692773 IC50 = 39300 nM T80975 CB1V6E 22692848 IC50 = 1020 nM T80975 CO2R3S 22692946 IC50 = 2100 nM T80975 C9WHT0 22692968 IC50 > 100000 nM T80975 CKB7C2 22693031 IC50 > 100000 nM T80975 C6CHV3 22693234 IC50 = 7790 nM T80975 CT39NL 22736235 IC50 = 85 nM T80975 C71MEZ 22971096 IC50 = 1900 nM T80975 COB60M 23133320 IC50 = 15 nM T80975 C9QLP0 23133323 IC50 = 40 nM T80975 C9VSU0 23141469 IC50 > 50000 nM T80975 C3F9LN 23366726 IC50 > 10000 nM T80975 C4QU3A 23366752 IC50 > 10000 nM T80975 CG12OL 23518511 IC50 = 500 nM T80975 C5AZ7B 23536770 IC50 = 7 nM T80975 CKID57 23589617 IC50 = 61 nM T80975 CRX0Q6 23625758 IC50 = 930 nM T80975 C0E2GY 23644614 IC50 > 10000 nM T80975 C56PGO 23644667 IC50 = 700 nM T80975 C7E0KL 23644828 IC50 = 1850 nM T80975 C4DBE2 23644829 IC50 > 10000 nM T80975 C72CKL 23644830 IC50 = 95 nM T80975 CC1TK5 23644831 IC50 = 3380 nM T80975 CLP8Y4 23644832 IC50 > 10000 nM T80975 C47NWC 23644833 IC50 = 1450 nM T80975 C2SG8A 23644834 IC50 > 10000 nM T80975 C0JRK8 23644835 IC50 = 2510 nM T80975 CKF20I 23644836 IC50 > 10000 nM T80975 CI64QY 23644837 IC50 = 1610 nM T80975 CL20MD 23644838 IC50 = 120 nM T80975 C4RW2C 23644839 IC50 = 1770 nM T80975 CK2HX6 23644840 IC50 = 15 nM T80975 CM0KD3 23644841 IC50 = 85 nM T80975 CS5HY0 23644842 IC50 > 10000 nM T80975 C4DFA5 23644843 IC50 = 560 nM T80975 CJ07AS 23644844 IC50 > 10000 nM T80975 CWQX87 23644845 IC50 = 3680 nM T80975 CP3L6Q 23644846 IC50 = 710 nM T80975 C9ATK1 23644847 IC50 = 1250 nM T80975 C8U6BV 23644848 IC50 = 93 nM T80975 CIZG50 23644849 IC50 = 2120 nM T80975 CKL39U 23644850 IC50 = 190 nM T80975 C4AEC8 23644851 IC50 = 1660 nM T80975 C47LSD 23644852 IC50 = 230 nM T80975 CT4XY0 23644853 IC50 = 330 nM T80975 CG48KV 23644854 IC50 = 860 nM T80975 C1JM4P 23644855 IC50 = 1080 nM T80975 CU90AF 23644856 IC50 = 1920 nM T80975 C3ZBS6 23644857 IC50 > 10000 nM T80975 CQI9A3 23644858 IC50 = 64 nM T80975 CM7C6T 23644859 IC50 = 560 nM T80975 CCI2M1 23644860 IC50 = 2540 nM T80975 C3Q5FV 23644861 IC50 > 10000 nM T80975 CR83MY 23644862 IC50 > 10000 nM T80975 CCI62P 23644863 IC50 > 10000 nM T80975 CHA4J3 23644864 IC50 > 10000 nM T80975 CB2C4G 23644865 IC50 > 10000 nM T80975 C9O4XE 23644866 IC50 > 10000 nM T80975 C5OQ2T 23644867 IC50 = 3870 nM T80975 C2WAK8 23644868 IC50 > 10000 nM T80975 C21APY 23644869 IC50 = 5640 nM T80975 CA92DC 23644870 IC50 = 380 nM T80975 CZ9L7X 23644871 IC50 > 10000 nM T80975 CK42DF 23644872 IC50 = 43 nM T80975 CO06PR 23644873 IC50 = 190 nM T80975 CH4S6V 23644874 IC50 = 250 nM T80975 CY9FT0 23644875 IC50 = 310 nM T80975 CEB43Q 23644876 IC50 > 10000 nM T80975 C2RN3L 23644877 IC50 = 44 nM T80975 C5XWJ8 23644878 IC50 = 44 nM T80975 CAZL79 23644879 IC50 = 58 nM T80975 CJR51Z 23644880 IC50 = 220 nM T80975 CGBW01 23644881 IC50 = 350 nM T80975 CUIT84 23644882 IC50 = 290 nM T80975 CZH4Q1 23644883 IC50 = 440 nM T80975 C3Y5BN 23644884 IC50 = 360 nM T80975 CSOG87 23644885 IC50 = 440 nM T80975 CT81BV 23644886 IC50 = 110 nM T80975 CM9YD6 23644887 IC50 = 860 nM T80975 CW20PU 23644888 IC50 = 550 nM T80975 C2ODX8 23644889 IC50 = 770 nM T80975 C9C5LQ 23644890 IC50 = 170 nM T80975 C7BGR4 23644891 IC50 > 10000 nM T80975 C6P1JN 23644892 IC50 > 10000 nM T80975 CIJ3K8 23644893 IC50 = 94 nM T80975 CV2MF6 23644894 IC50 = 67 nM T80975 CET2G3 23644895 IC50 = 87 nM T80975 CPX58K 23644896 IC50 = 85 nM T80975 C3U9RZ 23644897 IC50 = 2630 nM T80975 C3VPB8 23646046 IC50 = 1588 nM T80975 CSM47N 23646047 IC50 = 146 nM T80975 CT89CD 23646048 IC50 = 1189 nM T80975 CRF4T1 23646049 IC50 = 146 nM T80975 C2HYO8 23646050 IC50 = 1038 nM T80975 CS93DE 23646051 IC50 = 117 nM T80975 CV36WX 23646052 IC50 = 121 nM T80975 CT8CM3 23646053 IC50 = 43 nM T80975 CV63QL 23646054 IC50 = 115 nM T80975 C5W1PI 23646055 IC50 = 52 nM T80975 C9WDX0 23646056 IC50 = 52 nM T80975 C3P6TW 23646057 IC50 = 413 nM T80975 CQ95WB 23646058 IC50 = 201 nM T80975 CJ6VA1 23646059 IC50 = 93 nM T80975 C2EC7S 23646060 IC50 = 187 nM T80975 C0RG3C 23646061 IC50 = 214 nM T80975 CXT2S0 23646062 IC50 = 39 nM T80975 C7RJ3O 23646063 IC50 = 101 nM T80975 C1Q6OV 23646064 IC50 = 24 nM T80975 CXC16Y 23646065 IC50 = 62 nM T80975 C2PL8F 23646066 IC50 = 33 nM T80975 CYE8I2 23646067 IC50 = 44 nM T80975 CDE98J 23646068 IC50 = 11 nM T80975 C96KQX 23646931 IC50 > 8000 nM T80975 C6UJ1B 23646932 IC50 = 2000 nM T80975 C2MJ3D 23646933 IC50 = 675 nM T80975 C8YL1K 23646935 IC50 = 97 nM T80975 C3JWK1 23654166 IC50 = 300 nM T80975 CI6C1R 23658582 IC50 = 353 nM T80975 C6O8QY 23661616 IC50 = 2.7 nM T80975 C2S5ZM 23661662 Ki = 300 nM T80975 CYWG82 23729145 IC50 > 1000 nM T80975 CS2XY6 23817958 Ki = 103 nM T80975 C5LH1Q 23995100 IC50 = 2700 nM T80975 CARB19 24177555 Ki = 25 nM T80975 C2RV3U 24180608 IC50 = 1500 nM T80975 C5EX0A 24737647 IC50 = 1.3 nM T80975 C3X1WH 24742411 IC50 = 10 nM T80975 CS78XJ 24742412 IC50 = 150 nM T80975 C2KA6G 24742584 IC50 = 8 nM T80975 CN9GC8 24742586 IC50 = 25 nM T80975 CA3I4T 24753787 IC50 > 50000 nM T80975 CHU49V 24757938 IC50 = 0.03 nM T80975 C0D2PA 24758868 IC50 > 10000 nM T80975 C3K5YO 24758982 IC50 = 4066 nM T80975 CYU0Z8 24758983 IC50 = 4282 nM T80975 CJL67N 24759089 IC50 = 10990 nM T80975 C2APK8 24759090 IC50 > 10000 nM T80975 C5CRF6 24759091 IC50 = 3954 nM T80975 CA8U7X 24759094 IC50 = 515 nM T80975 CRB89L 24759205 IC50 = 1624 nM T80975 C13JUP 24759314 IC50 > 10000 nM T80975 C7YG1N 24759534 IC50 < 10 nM T80975 CAJ4T2 24762205 IC50 = 4233 nM T80975 CQNP54 24764449 IC50 = 1000 nM T80975 CCPS81 24764502 IC50 > 35000 nM T80975 CJ52YI 24765042 IC50 = 9 nM T80975 C2UOE0 24766030 IC50 > 50000 nM T80975 CMP4F2 24767979 IC50 = 1.1 nM T80975 CCF17D 24768394 IC50 = 18840 nM T80975 CYK71D 24768395 IC50 > 12500 nM T80975 C7EXG0 24768396 IC50 > 12500 nM T80975 C4Z9CN 24769780 Ki = 83 nM T80975 CJUK39 24770517 IC50 > 10000 nM T80975 C81GVC 24774737 IC50 = 79.43 nM T80975 CN6B1L 24774912 IC50 = 794.33 nM T80975 CP9G0L 24783392 IC50 = 1480 nM T80975 C9PA0M 24807809 IC50 > 10000 nM T80975 C0JUN4 24812717 IC50 = 48 nM T80975 CP6N9M 24812718 IC50 > 25000 nM T80975 CW0G8H 24812719 IC50 > 5000 nM T80975 CSM5E4 24822265 IC50 = 7 nM T80975 CA80DO 24822266 IC50 = 45.71 nM T80975 CHL9K0 24822267 IC50 = 4 nM T80975 CF3TD8 24822268 IC50 = 0.2 nM T80975 CL3GM9 24822269 IC50 = 1 nM T80975 C0B7TO 24822426 IC50 = 0.5 nM T80975 C6P1OH 24822427 IC50 = 2 nM T80975 C24UQW 24822428 IC50 = 0.7943 nM T80975 CROH43 24822429 IC50 = 1.995 nM T80975 CT48RV 24822430 IC50 = 0.8 nM T80975 CO9Z0H 24822598 IC50 = 10.96 nM T80975 C51IZL 24822599 IC50 = 12.02 nM T80975 CA90EF 24822600 IC50 = 5.495 nM T80975 CYL8J4 24822601 IC50 = 22.91 nM T80975 CDX96O 24822602 IC50 > 1400 nM T80975 C2MUA7 24823072 IC50 = 530 nM T80975 CX94DT 24823073 IC50 = 1900 nM T80975 C4A6LB 24823090 IC50 = 15 nM T80975 C2B4JP 24823091 IC50 = 1500 nM T80975 CF6M3W 24823093 IC50 = 2.884 nM T80975 C0NLO8 24823094 IC50 = 1.3 nM T80975 C7D8PC 24823095 IC50 = 1.2 nM T80975 C14FLQ 24823250 IC50 = 3.8 nM T80975 C3KPO7 24823251 IC50 = 4.169 nM T80975 C36BFD 24823252 IC50 = 314 nM T80975 CBF60S 24823253 IC50 = 28 nM T80975 C3A2BF 24823416 IC50 > 25000 nM T80975 CYBI02 24823426 IC50 = 205 nM T80975 C45UGH 24823586 IC50 = 5 nM T80975 CFA3T8 24823588 IC50 = 3784 nM T80975 C51ZTV 24823589 IC50 = 1123 nM T80975 CX0QC1 24823590 IC50 = 54 nM T80975 CR7CH6 24823736 IC50 > 25000 nM T80975 C26KXV 24823738 IC50 = 2540 nM T80975 CO3K7R 24823740 IC50 = 13 nM T80975 CJ5N0F 24823896 IC50 = 3 nM T80975 CBLJ48 24823898 IC50 > 5000 nM T80975 CI5HZ0 24824043 IC50 = 18.2 nM T80975 C6AI4Q 24824044 IC50 = 310 nM T80975 C0OW9S 24824045 IC50 = 19.95 nM T80975 CG0K1Z 24824046 IC50 > 8300 nM T80975 CDT3L2 24824050 IC50 = 1 nM T80975 CLN48F 24824051 IC50 = 3 nM T80975 C0NXE2 24824052 IC50 = 1 nM T80975 C7SU8H 24824183 IC50 = 28.18 nM T80975 CQS3X5 24824184 IC50 = 1 nM T80975 C1R5GU 24824185 IC50 = 19.95 nM T80975 C7Y2SE 24824186 IC50 = 1.995 nM T80975 C7T9FG 24824187 IC50 = 1.995 nM T80975 CWTI12 24824188 IC50 = 52.48 nM T80975 CQ1A8W 24824189 IC50 = 0.5 nM T80975 C8RE5C 24824190 IC50 = 25.7 nM T80975 C3K1FM 24824191 IC50 = 62 nM T80975 CG5VC7 24824313 IC50 = 0.6 nM T80975 CWG51N 24824314 IC50 = 0.302 nM T80975 CD93XN 24824315 IC50 = 0.3 nM T80975 CFI7E9 24824316 IC50 = 0.8 nM T80975 C6K5ST 24824317 IC50 = 0.302 nM T80975 CV0S5L 24824318 IC50 = 19.05 nM T80975 CUK14T 24824319 IC50 = 58 nM T80975 CZ09ID 24824320 IC50 = 39.81 nM T80975 CM28KX 24824321 IC50 = 40 nM T80975 CD57UN 24824322 IC50 = 25.7 nM T80975 CNI50G 24824323 IC50 = 40 nM T80975 C9ERB8 24824446 IC50 = 0.6 nM T80975 CGDB50 24824447 IC50 = 1 nM T80975 C84VZK 24824448 IC50 = 1.3 nM T80975 C6OC4K 24824449 IC50 = 1.288 nM T80975 CLU56Y 24824450 IC50 = 0.3 nM T80975 CO71SC 24824451 IC50 = 21.88 nM T80975 C5BA7V 24824452 IC50 = 0.6 nM T80975 CR49SP 24824453 IC50 = 77.62 nM T80975 CG64EL 24824454 IC50 = 95 nM T80975 CTH69P 24824602 IC50 = 8 nM T80975 CQN3Z7 24825710 IC50 = 1490 nM T80975 CS1B9V 24849200 IC50 = 1 nM T80975 CX0S9L 24854902 IC50 = 505 nM T80975 C1SVT2 24854903 IC50 = 2680 nM T80975 C61KPI 24856363 IC50 > 20000 nM T80975 CS82HN 24856408 IC50 = 2200 nM T80975 CZ5Y4H 24856498 IC50 = 3400 nM T80975 CALJ74 24859856 IC50 = 49 nM T80975 CCS58O 24863072 IC50 = 230 nM T80975 C6C2GX 24863500 IC50 = 170 nM T80975 CYVB83 24863584 IC50 = 420 nM T80975 CQ15ML 24863670 IC50 = 240 nM T80975 C4XZ3N 24863671 IC50 > 25000 nM T80975 CE3IW4 24879184 IC50 > 5000 nM T80975 C7V8BA 24879242 IC50 > 5000 nM T80975 CT76XV 24879243 IC50 = 4300 nM T80975 CGD8J5 24879244 IC50 > 5000 nM T80975 C1XWO7 24879245 IC50 = 3400 nM T80975 CA21RX 24879305 IC50 = 1400 nM T80975 COF05N 24879306 IC50 > 1000 nM T80975 C6NIQ2 24879307 IC50 = 11 nM T80975 C45HIT 24879308 IC50 = 1800 nM T80975 CM6G7A 24879309 IC50 > 5000 nM T80975 C0KW5Y 24879310 IC50 > 5000 nM T80975 C7M9FB 24879311 IC50 > 5000 nM T80975 C0ZJX6 24879366 IC50 > 5000 nM T80975 C5NA4Z 24879367 IC50 = 4400 nM T80975 CDJE41 24879368 IC50 > 5000 nM T80975 C4MG3B 24882476 IC50 = 255 nM T80975 CFK2B9 24882503 IC50 = 960 nM T80975 C43HWQ 24883287 IC50 = 1300 nM T80975 C8DA5Q 24883334 IC50 = 600 nM T80975 CRB0L1 24884602 IC50 = 27 nM T80975 COY07V 24884826 IC50 = 19 nM T80975 C0P6AU 24894017 IC50 = 818 nM T80975 C4V9GH 24894117 IC50 = 31 nM T80975 CJ4V1O 24894180 IC50 = 72 nM T80975 C7DU4K 24894181 IC50 = 810 nM T80975 C4AKV2 24894182 IC50 > 12500 nM T80975 CG78MT 24894183 IC50 = 74 nM T80975 C0NTK9 24894184 IC50 = 14 nM T80975 CTJ4X5 24894299 IC50 = 2000 nM T80975 CHJ9E0 24894300 IC50 > 12500 nM T80975 C1KDM0 24894301 IC50 = 6600 nM T80975 C5P7AU 24894302 IC50 = 10000 nM T80975 CY64PL 24894303 IC50 = 3500 nM T80975 CLSZ06 24894406 IC50 = 11 nM T80975 C39BFI 24894407 IC50 = 17 nM T80975 C3E7OF 24894408 IC50 = 9 nM T80975 C9OF4S 24894409 IC50 = 930 nM T80975 C24JVL 24894410 IC50 = 790 nM T80975 CE52TC 24894505 IC50 = 6100 nM T80975 C34HBJ 24894506 IC50 = 39 nM T80975 CR70JM 24894507 IC50 > 12500 nM T80975 CYP89A 24894508 IC50 > 12500 nM T80975 CGI19K 24894509 IC50 = 47 nM T80975 C4RG3F 24894510 IC50 = 17 nM T80975 CFPQ62 24894511 IC50 > 12500 nM T80975 CZ9CN1 24894618 IC50 = 15 nM T80975 C5E2ZL 24894619 IC50 = 33 nM T80975 CVH87X 24894620 IC50 = 1 nM T80975 C58YJN 24894621 IC50 = 25 nM T80975 CR47VO 24894622 IC50 = 100 nM T80975 C53BYS 24894623 IC50 = 500 nM T80975 CS4F6K 24894763 IC50 > 12500 nM T80975 CKE29C 24894764 IC50 = 1600 nM T80975 CW3IF0 24894765 IC50 = 44 nM T80975 CM6K3X 24894768 IC50 = 5900 nM T80975 CJH19T 24894883 IC50 = 15000 nM T80975 CJ14YB 24894884 IC50 = 13000 nM T80975 CHVU39 24894885 IC50 = 31000 nM T80975 CZ6KD4 24894886 IC50 = 3100 nM T80975 CKBY19 24894887 IC50 = 2300 nM T80975 C57BHF 24894888 IC50 = 5300 nM T80975 CB5TP8 24894992 IC50 = 4400 nM T80975 C32SUJ 24894993 IC50 = 1600 nM T80975 C38TGD 24894994 IC50 = 8000 nM T80975 CP7QT2 24894995 IC50 = 11000 nM T80975 C41SIT 24894996 IC50 = 5200 nM T80975 CFW40U 24894997 IC50 = 1500 nM T80975 CF4N9X 24895100 IC50 = 4200 nM T80975 CDR4Q6 24895757 IC50 > 12500 nM T80975 CN13JF 24899915 IC50 = 0.7 ug.mL-1 T80975 CBWR97 24899916 IC50 = 0.64 ug.mL-1 T80975 C9F2JD 24899917 IC50 > 10 ug.mL-1 T80975 C64MTI 24900160 IC50 = 3.8 ug.mL-1 T80975 CO2I6Q 24900161 IC50 = 5.1 ug.mL-1 T80975 CD08VO 24901691 Ki = 23.7 nM T80975 C0NCI3 24901692 IC50 = 329 nM T80975 C59ICM 24901693 IC50 = 236 nM T80975 C9WD7I 24901694 IC50 = 208 nM T80975 C9KJD4 24901695 Ki = 2 nM T80975 C6UXO8 24901699 IC50 = 1134 nM T80975 C34BSE 24901700 IC50 = 346 nM T80975 C2CD9F 24901701 IC50 = 127 nM T80975 CN9W4J 24901702 IC50 = 90 nM T80975 CVAC46 24901703 IC50 = 344 nM T80975 CNK14W 24901705 IC50 = 11 nM T80975 CAN86I 24901706 IC50 = 25 nM T80975 C58CHD 24901707 IC50 = 25 nM T80975 C0UM9A 24901708 IC50 = 28 nM T80975 CSCB80 24901709 IC50 = 17 nM T80975 C6PDE3 24901710 IC50 = 113 nM T80975 C2KI4J 24901711 IC50 = 94 nM T80975 C2UWO4 24901712 IC50 = 145 nM T80975 CF0KV6 24901713 IC50 = 32 nM T80975 CJO43A 24901714 IC50 = 31 nM T80975 C6OAM7 24901715 IC50 = 593 nM T80975 CIH4C8 24901716 IC50 = 175 nM T80975 CB79YC 24905143 IC50 = 213 nM T80975 C2DC9J 24905144 IC50 = 1100 nM T80975 CN6V8Z 24905145 IC50 = 55 nM T80975 CSB7P5 24905148 IC50 > 50000 nM T80975 CGSF21 24905149 IC50 > 50000 nM T80975 CVDG02 24905150 IC50 = 2230 nM T80975 CWH6C5 24905152 IC50 = 310 nM T80975 C0HE2Q 24905153 IC50 = 7000 nM T80975 C7QSC9 24905154 IC50 = 1680 nM T80975 CO9D0K 24905155 IC50 = 100000 nM T80975 C5W9UR 24905157 IC50 = 1050 nM T80975 CC1DA3 24905158 IC50 = 1020 nM T80975 COW79F 24905159 IC50 = 100000 nM T80975 CFPA53 24905160 IC50 = 43000 nM T80975 C2O0JX 24905161 IC50 = 5890 nM T80975 CA72BE 24905162 IC50 = 4600 nM T80975 CQN6X9 24905163 IC50 = 1640 nM T80975 CD4O1F 24905165 IC50 = 100000 nM T80975 CKL48T 24905166 IC50 = 11000 nM T80975 C76VYL 24905167 IC50 = 4800 nM T80975 C7K5PU 24905168 IC50 = 4360 nM T80975 CZ57ID 24905169 IC50 = 100000 nM T80975 C2DHX9 24905170 IC50 = 100000 nM T80975 CSB96E 24905171 IC50 = 100000 nM T80975 CWZ0R2 24905172 IC50 = 21000 nM T80975 CY3B6M 24905175 IC50 = 100000 nM T80975 CW7UA3 24905176 IC50 = 3120 nM T80975 CW1V0H 24905177 IC50 = 100000 nM T80975 CO6Y0L 24905178 IC50 = 5290 nM T80975 C4MO8B 24905180 IC50 = 1660 nM T80975 COJI47 24905181 IC50 = 901 nM T80975 CS0B2C 24905182 IC50 = 48 nM T80975 C1H4BT 24905183 IC50 = 752 nM T80975 C4WHK9 24905184 IC50 = 1020 nM T80975 C7Q4MZ 24905185 IC50 = 153 nM T80975 CS4IP1 24905186 IC50 = 44 nM T80975 C69QWO 24905187 IC50 = 840 nM T80975 C85ANB 24905188 IC50 = 76 nM T80975 CNHD75 24905189 IC50 = 1690 nM T80975 C9JUO2 24905190 IC50 = 6900 nM T80975 CPR03K 24905191 IC50 = 4130 nM T80975 CTAG19 24905193 IC50 = 9 nM T80975 C7VJM5 24905194 IC50 = 100000 nM T80975 CEP1L3 24905195 IC50 = 2900 nM T80975 CP68ZD 24905196 IC50 = 1220 nM T80975 C8Z0RJ 24905197 IC50 = 109 nM T80975 CN9RT0 24905198 IC50 = 194 nM T80975 CHI78P 24905200 IC50 = 5600 nM T80975 CO6PE8 24905201 IC50 = 470 nM T80975 CZ63HS 24905202 IC50 = 19 nM T80975 C2X0FC 24905203 IC50 = 420 nM T80975 C0WCE3 24905204 IC50 = 12000 nM T80975 CNK50B 24905205 IC50 = 4400 nM T80975 C12DPB 24905206 IC50 = 330 nM T80975 C8N0RH 24905207 IC50 = 550 nM T80975 CYA5G2 24905208 IC50 = 1100 nM T80975 CDV2B4 24905209 IC50 = 11000 nM T80975 CEFK68 24905210 IC50 = 940 nM T80975 CUFP12 24905211 IC50 = 1600 nM T80975 C0JG8L 24905212 IC50 = 134 nM T80975 CQ13ZI 24905215 IC50 = 49000 nM T80975 C6VI8F 24905216 IC50 = 960 nM T80975 CXNH25 24905217 IC50 = 19000 nM T80975 C2PN9S 24905218 IC50 = 13000 nM T80975 C9O2AL 24905219 IC50 = 100000 nM T80975 CIT7U8 24905220 IC50 = 100000 nM T80975 CMD26S 24905221 IC50 = 715 nM T80975 C4R8WC 24905222 IC50 = 172 nM T80975 C47SHA 24905223 IC50 = 295 nM T80975 C1DY2R 24905224 IC50 = 411 nM T80975 CS0XF9 24905225 IC50 = 12000 nM T80975 CG5VX2 24905226 IC50 = 100000 nM T80975 C57QEO 24905227 IC50 = 100000 nM T80975 C7CG5E 24905228 IC50 = 50000 nM T80975 CHP5D1 24905229 IC50 = 100000 nM T80975 CXP09S 24905230 IC50 = 14000 nM T80975 CY7XG1 24905231 IC50 = 100000 nM T80975 C7JFQ2 24905232 IC50 = 5100 nM T80975 C2JM1P 24905233 IC50 = 7000 nM T80975 CC3BF0 24905234 IC50 = 100000 nM T80975 CE57FI 24905235 IC50 = 1400 nM T80975 CUP20O 24905236 IC50 = 4300 nM T80975 CLC6Q2 24905237 IC50 = 100000 nM T80975 C9M1GI 24905238 IC50 = 1200 nM T80975 CVD72F 24905239 IC50 = 6300 nM T80975 CK38IZ 24905240 IC50 = 1400 nM T80975 CO2V5E 24905241 IC50 = 13000 nM T80975 CZBA19 24905244 IC50 = 215 nM T80975 CQ8OI1 24905246 IC50 = 100000 nM T80975 CIF2J5 24905251 IC50 = 2600 nM T80975 CPTE58 24905252 IC50 = 2160 nM T80975 CP50RD 24905280 IC50 = 68 nM T80975 CG13ZM 24905281 IC50 = 566 nM T80975 CF0S6X 24905282 IC50 = 13400 nM T80975 C5HBL0 24905284 IC50 = 100000 nM T80975 C2Z5DN 24905285 IC50 = 237 nM T80975 CL6GH8 24905286 IC50 = 1060 nM T80975 CKYO98 24905287 IC50 = 10 nM T80975 CRNQ65 24905288 IC50 = 119 nM T80975 COD7I5 24905289 IC50 = 43 nM T80975 C4LP7E 24905290 IC50 = 151 nM T80975 C2GI1R 24905292 IC50 = 100000 nM T80975 CHW8C4 24905293 IC50 = 279 nM T80975 CQF0H1 24905294 IC50 = 259 nM T80975 CNO7X0 24905295 IC50 = 20 nM T80975 C5WRG7 24905296 IC50 = 2070 nM T80975 CQ1S0U 24905297 IC50 = 100000 nM T80975 C4UES7 24905298 IC50 = 100000 nM T80975 CMS69P 24905299 IC50 = 7160 nM T80975 CC0U5M 24905300 IC50 = 4.3 nM T80975 CW7X6S 24905301 IC50 = 11800 nM T80975 C97IQV 24905302 IC50 = 106 nM T80975 CSJ47V 24905303 IC50 = 3780 nM T80975 CPN74C 24905304 IC50 = 3120 nM T80975 C5CS3N 24905305 IC50 = 435 nM T80975 CK4XE9 24905307 IC50 = 100000 nM T80975 CTU6Z3 24905308 IC50 = 100000 nM T80975 C9SQX1 24905309 IC50 = 369 nM T80975 CM75JP 24905310 IC50 = 1750 nM T80975 C9Q2BJ 24905311 IC50 = 872 nM T80975 C9VUA1 24905312 IC50 = 174 nM T80975 CU3RS1 24905313 IC50 = 1150 nM T80975 CYG3H2 24905314 IC50 = 1150 nM T80975 CV5Q7O 24905315 IC50 = 77 nM T80975 C8SA3O 24905316 IC50 = 55 nM T80975 CI5MN3 24905317 IC50 = 66 nM T80975 CJ1P7K 24905318 IC50 = 103 nM T80975 C1T6YQ 24905319 IC50 = 401 nM T80975 CAU86X 24905320 IC50 = 555 nM T80975 C54ISY 24905321 IC50 = 1900 nM T80975 C2GE5I 24905322 IC50 = 554 nM T80975 C8D6YK 24905323 IC50 = 2800 nM T80975 C5NZH9 24905324 IC50 = 1140 nM T80975 C9D6JR 24905325 IC50 = 517 nM T80975 CLZT41 24905326 IC50 = 62 nM T80975 CW8FD3 24905327 IC50 = 178 nM T80975 CHB7A2 24905328 IC50 = 2130 nM T80975 CA8EI3 24905329 IC50 = 2900 nM T80975 CCQ0O7 24905330 IC50 = 100000 nM T80975 CJ81AS 24905331 IC50 = 3000 nM T80975 C8PW4H 24905332 IC50 = 40 nM T80975 C2Y5TF 24905333 IC50 = 55 nM T80975 CH9FL5 24905334 IC50 = 10000 nM T80975 C1S0PC 24905335 IC50 = 100000 nM T80975 C8N9MV 24905336 IC50 = 2020 nM T80975 C9E8BJ 24905338 IC50 = 98800 nM T80975 CX85AC 24905341 IC50 = 100000 nM T80975 CKZ80E 24905342 IC50 = 93 nM T80975 CO8SH1 24905343 IC50 = 100000 nM T80975 C7IZL6 24905344 IC50 = 100000 nM T80975 CUIG07 24905422 IC50 = 230 nM T80975 CJRU52 24936082 IC50 = 700 nM T80975 C5ZM4T 24936119 IC50 > 10000 nM T80975 C8DG1Y 24941253 IC50 > 10000 nM T80975 CB3L5X 24949544 IC50 = 1.7 nM T80975 CC4K1P 24949545 IC50 = 36 nM T80975 C17QKF 24949548 IC50 = 7.6 nM T80975 C39STN 24949698 IC50 = 6.3 nM T80975 CCA9G2 24949700 IC50 = 5.6 nM T80975 CFU0T1 24949702 IC50 = 2.6 nM T80975 CE79PI 24949704 IC50 = 63 nM T80975 C15BZP 24949852 IC50 = 2100 nM T80975 CZHE50 24949856 IC50 = 8600 nM T80975 CJ0IO9 24958482 IC50 = 8 nM T80975 CSI2X7 24958841 IC50 = 4 nM T80975 C30ILA 24959937 IC50 = 18 nM T80975 CUAD69 24959938 IC50 = 165 nM T80975 CHQZ58 24959939 IC50 = 92 nM T80975 C2VTM7 24960306 IC50 = 225 nM T80975 C6G8MR 24960307 IC50 = 3000 nM T80975 CU2S7R 24960308 IC50 = 1 nM T80975 C7BD9Z 24960309 IC50 = 3 nM T80975 C2TR9I 24960310 IC50 = 1 nM T80975 C29ACE 24960670 IC50 = 13 nM T80975 CN9QH4 24960671 IC50 = 8 nM T80975 C6PU3R 24960672 IC50 = 2 nM T80975 CZR85I 24960673 IC50 = 3 nM T80975 CU7I2E 24963046 IC50 = 10.5 nM T80975 C9JB2R 24966651 IC50 = 30 nM T80975 C4RGC1 24967005 IC50 = 360 nM T80975 CTDN38 24967006 IC50 = 30 nM T80975 C9YN2Q 24967131 IC50 > 10000 nM T80975 CD5HQ0 24969301 IC50 > 10000 nM T80975 CT8OF0 24983254 IC50 = 30 nM T80975 CVF62Q 24983255 IC50 = 88 nM T80975 CX6FR3 24983298 IC50 = 6358 nM T80975 CEQ1F2 24983299 IC50 = 2059 nM T80975 C6JXE2 24983340 IC50 = 6000 nM T80975 CK9TP6 24983359 IC50 > 25000 nM T80975 CC39KU 24983384 IC50 > 25000 nM T80975 C07PXL 24983399 IC50 > 25000 nM T80975 C03XEW 24983494 IC50 = 1570 nM T80975 CQ46VT 24983495 IC50 = 1380 nM T80975 C4EG8R 24993189 IC50 > 10000 nM T80975 CS3Q8B 24995659 Ki > 4000 nM T80975 CBK82P 25011729 IC50 > 30000 nM T80975 CN3FQ5 25014760 IC50 = 100 nM T80975 C3WX2S 25014762 IC50 = 94 nM T80975 COB43M 25014810 IC50 = 3200 nM T80975 C3SE8L 25014843 IC50 = 27 nM T80975 CV0RN4 25014844 IC50 = 141 nM T80975 CZ8LP3 25014846 IC50 = 115 nM T80975 CO0R9B 25014936 IC50 = 965 nM T80975 CRA79I 25015025 IC50 = 22 nM T80975 CGDP84 25015026 IC50 = 190 nM T80975 CSD14Z 25015027 IC50 = 589 nM T80975 C0HVE3 25015107 IC50 = 231 nM T80975 CV67GQ 25015556 IC50 = 390 nM T80975 CRO0Y8 25022735 IC50 > 200000 nM T80975 C72AJM 25022736 IC50 > 200000 nM T80975 CI7ZE2 25023830 IC50 = 460 nM T80975 CB38WD 25027538 IC50 > 400000 ug.mL-1 T80975 CY0Q5S 25027755 IC50 > 400000 ug.mL-1 T80975 C6PKS5 25028418 IC50 > 400000 ug.mL-1 T80975 CS0P4K 25054599 IC50 = 10 nM T80975 C2F1YJ 25054600 IC50 = 210 nM T80975 C0UDM4 25054601 IC50 = 20 nM T80975 C8CA3Y 25054857 IC50 = 1400 nM T80975 CDYM40 25055101 IC50 > 10000 nM T80975 CMH4W3 25055102 IC50 = 2000 nM T80975 CQZ95L 25055103 IC50 = 1400 nM T80975 C8UGB1 25055104 IC50 = 700 nM T80975 CAE17C 25055344 IC50 = 800 nM T80975 CHLQ49 25063262 IC50 > 100000 nM T80975 C2KY1G 25094210 IC50 = 36 nM T80975 CMD8J5 25094492 IC50 = 475 nM T80975 C1G5IO 25094493 IC50 = 51 nM T80975 COS3T6 25094494 IC50 = 206 nM T80975 CH90KV 25097876 IC50 = 39 nM T80975 C9L5ID 25098154 IC50 = 130 nM T80975 C1DYP9 25098155 IC50 = 203 nM T80975 C9P1IU 25098159 IC50 = 718 nM T80975 C53XHG 25098428 IC50 = 389 nM T80975 CAO38V 25098429 IC50 = 16 nM T80975 C7FI3O 25098430 IC50 = 102 nM T80975 CMB52V 25098432 IC50 = 70 nM T80975 C2P0EV 25102846 IC50 = 3 nM T80975 CS96TK 25113168 IC50 = 34 nM T80975 CQ27UI 25113814 IC50 = 90 nM T80975 C2IHY0 25114266 IC50 = 1 nM T80975 CP8S9W 25116064 IC50 = 26 nM T80975 CTV54O 25123227 IC50 = 0.26 nM T80975 C1IYN7 25127854 IC50 = 1.1 nM T80975 CKD14B 25127856 IC50 = 1.1 nM T80975 C3OV0B 25127857 IC50 = 1.9 nM T80975 CJBX60 25128180 IC50 = 1.3 nM T80975 CC5SD9 25128181 IC50 = 3.6 nM T80975 CF7C5B 25129829 IC50 = 5145 nM T80975 CXNM84 25129830 IC50 = 3042 nM T80975 CY2S1P 25129831 IC50 > 10000 nM T80975 CQMU82 25138148 IC50 = 6 nM T80975 CD9O6K 25138149 IC50 = 169 nM T80975 CGT1W6 25144294 IC50 = 4 nM T80975 CU7VR0 25144732 IC50 <= 1 nM T80975 C6BWZ8 25145145 IC50 = 550 nM T80975 CSO82D 25154877 Ki = 1590 nM T80975 CB21XV 25164469 Ki = 3978 nM T80975 CNF0A8 25164674 Ki > 8880 nM T80975 CUX83H 25164675 Ki > 8880 nM T80975 C1H7BF 25164677 Ki > 8880 nM T80975 CN50EI 25164678 Ki > 8880 nM T80975 C3XI7P 25164880 Ki > 8880 nM T80975 CX80QK 25164883 Ki > 8880 nM T80975 C6SD2A 25165081 Ki > 8880 nM T80975 C67TVH 25165085 Ki > 8880 nM T80975 C8J4KL 25165278 Ki = 3291 nM T80975 CRJ6M7 25165279 Ki > 8880 nM T80975 C7RBX0 25165280 Ki > 8880 nM T80975 CPEY29 25165481 Ki > 8880 nM T80975 C70DRX 25165482 Ki > 8880 nM T80975 CE8D1W 25165860 Ki = 3554 nM T80975 C6VZU2 25165861 Ki > 8880 nM T80975 CVI70X 25166053 Ki > 915 nM T80975 C9VA1N 25166056 Ki > 915 nM T80975 C5BM7F 25166250 Ki = 13142 nM T80975 CCN25J 25166251 Ki = 2710 nM T80975 C1CNX7 25166659 Ki = 126500 nM T80975 C81WIV 25166867 Ki > 915 nM T80975 C9MR2O 25166869 Ki = 5339 nM T80975 CF4G1L 25167074 Ki > 8880 nM T80975 C35ZXL 25167075 Ki > 8880 nM T80975 C1CRJ7 25167076 Ki > 8880 nM T80975 C1IFX5 25167077 Ki > 8880 nM T80975 C2D3FP 25167078 Ki > 8880 nM T80975 CP2W8I 25167079 Ki > 8880 nM T80975 CJO5A4 25167275 Ki > 8880 nM T80975 C5KX0G 25167277 Ki > 8880 nM T80975 CQ5FJ8 25167278 Ki > 8880 nM T80975 C37YSX 25167280 Ki > 8880 nM T80975 CX0O5A 25178331 IC50 = 4300 nM T80975 CIG4H0 25178539 IC50 = 4100 nM T80975 COB9G8 25181586 IC50 = 22600 nM T80975 C76WYH 25184035 IC50 = 430 nM T80975 CTED51 25186142 IC50 = 125.89 nM T80975 C8YLD6 25194331 IC50 = 130 nM T80975 CXC9B3 25194865 IC50 = 1000 nM T80975 C1I0VS 25194866 IC50 = 190 nM T80975 C9OZN3 25194867 IC50 = 5300 nM T80975 CPQ31L 25195294 IC50 = 214.7 nM T80975 CYK1V8 25206185 IC50 = 2.8 nM T80975 C6FGQ1 25206346 IC50 = 1.2 nM T80975 C8ZBN0 25206349 IC50 = 64 nM T80975 CXNW87 25207322 IC50 = 1 nM T80975 CNG96H 25210579 IC50 > 10000 nM T80975 CRO09K 25211064 IC50 = 1000 nM T80975 CNQ9G5 25218180 IC50 < 1000 nM T80975 C8IJB9 25218207 IC50 = 56300 nM T80975 C6I9ND 25231072 IC50 = 119 nM T80975 CEM5K4 25256719 IC50 = 309 nM T80975 CRO8T9 25263033 Ki > 12500 nM T80975 C4AR9G 25268137 IC50 = 2500 nM T80975 CLB28U 25271180 IC50 > 100000 nM T80975 CGHR32 25271181 IC50 > 100000 nM T80975 C3E9XU 25271513 IC50 > 100000 nM T80975 CGBX14 25271514 IC50 > 100000 nM T80975 C76NWM 25271515 IC50 > 100000 nM T80975 C6C4YR 25271516 IC50 > 100000 nM T80975 CUAK50 25271517 IC50 > 100000 nM T80975 CIR67H 25271518 IC50 > 100000 nM T80975 CE1L2V 29786650 IC50 = 3.8 nM T80975 CUJB21 32402967 IC50 = 753 nM T80975 CN46JI 36217989 IC50 > 1000 nM T80975 C8T5IH 42602949 IC50 = 398.11 nM T80975 C41TLH 42603880 IC50 = 81000 nM T80975 CS1AT2 42603881 IC50 = 58000 nM T80975 CZ2VH7 42604008 IC50 = 30000 nM T80975 C81UIT 42604010 IC50 = 25000 nM T80975 CU2B4F 42611245 IC50 = 37 nM T80975 C7GIQ3 42625508 IC50 = 9200 nM T80975 CVZ83M 42625582 IC50 = 7800 nM T80975 C5MD9E 42625892 IC50 = 6100 nM T80975 C8B6TY 42628503 EC50 < 500 nM T80975 CJ5U1X 42639664 IC50 = 3.4 ug.mL-1 T80975 C0C1HL 42645248 IC50 = 989 nM T80975 CS3AI0 42645478 IC50 = 430 nM T80975 CM41UJ 43176565 IC50 = 26.5 nM T80975 CK76WN 43176566 IC50 = 9.6 nM T80975 CPS5F6 43517028 IC50 = 0.68 nM T80975 CAK0F2 44155856 IC50 = 15 nM T80975 CHQ24O 44156904 IC50 = 85 nM T80975 CI50DJ 44156905 Ki = 140 nM T80975 CNH12Z 44156906 IC50 = 140 nM T80975 C1V7TM 44156907 IC50 = 270 nM T80975 CT19KO 44156908 IC50 = 310 nM T80975 CTN41Y 44156909 IC50 = 3400 nM T80975 C2W0XB 44156915 Ki = 80 nM T80975 CN0X1C 44156917 IC50 > 10000 nM T80975 CIM89D 44157074 IC50 = 87 nM T80975 CLW80F 44160269 IC50 = 3800 nM T80975 CSH3D6 44177697 IC50 = 1200 nM T80975 C65VUH 44177803 IC50 = 40 nM T80975 CO6HU7 44178069 IC50 = 108 nM T80975 C9S7VY 44181153 IC50 = 3.4 nM T80975 CNJ3Y1 44181654 IC50 = 1300 nM T80975 CW7ZK4 44181971 IC50 = 31.2 nM T80975 CB0O2A 44186880 Ki > 8880 nM T80975 C9K7OP 44186882 Ki > 8880 nM T80975 CX0ZU8 44186885 Ki > 8880 nM T80975 CNGV37 44189584 Ki > 8880 nM T80975 C8KNA3 44219632 Ki > 4000 nM T80975 C0VIX4 44219633 Ki > 4000 nM T80975 CK73NR 44219749 IC50 > 50000 nM T80975 CN2QG1 44223357 IC50 = 4300 nM T80975 CEL61X 44229839 IC50 > 10000 nM T80975 C4NWP5 44246325 IC50 > 500000 nM T80975 C2EW0I 44246326 IC50 = 5000 nM T80975 CSD8T0 44246327 IC50 = 13700 nM T80975 CMKF08 44246328 IC50 > 500000 nM T80975 CAO87V 44246329 IC50 > 500000 nM T80975 CLU2V3 44246330 IC50 > 500000 nM T80975 C73CBF 44247727 IC50 = 30 nM T80975 CHZ6Q1 44269004 IC50 = 85 nM T80975 CSH9V7 44290834 IC50 = 892 nM T80975 CT2FY7 44291004 IC50 = 105 nM T80975 CJ0ED9 44291208 IC50 = 1808 nM T80975 CZFQ76 44291533 IC50 > 50000 nM T80975 CSD7V2 44299148 IC50 = 115 nM T80975 CH3J2E 44299176 IC50 = 60 nM T80975 C27GVO 44299203 IC50 = 100 nM T80975 CY6WC0 44299236 IC50 = 800 nM T80975 C3RG0C 44299304 IC50 = 500 nM T80975 CJM26I 44299321 IC50 = 7100 nM T80975 C9UGL3 44299325 IC50 = 300 nM T80975 CJEZ96 44299338 IC50 = 400 nM T80975 C8XGN5 44299339 IC50 = 300 nM T80975 CNH34G 44299354 IC50 = 400 nM T80975 C82MSD 44299360 IC50 = 2300 nM T80975 CEU2W4 44308690 IC50 = 270 nM T80975 CY6ZB5 44308830 IC50 = 2680 nM T80975 C1I6RG 44308968 IC50 = 161 nM T80975 C1I0LN 44308993 IC50 = 144 nM T80975 CKVZ38 44308994 IC50 = 129 nM T80975 CF9I2S 44309110 IC50 = 3680 nM T80975 C8VX1L 44309229 IC50 = 5060 nM T80975 CZQ4S0 44309230 IC50 = 29 nM T80975 CHF28G 44309494 IC50 = 6890 nM T80975 CQN1R8 44331899 IC50 = 3700 nM T80975 C1KSW5 44335197 IC50 > 1000 nM T80975 C0KD4U 44346053 IC50 = 1400 nM T80975 CYV2D7 44368815 IC50 = 9 nM T80975 CI3W6L 44378535 IC50 = 17 nM T80975 C5M3ZC 44382107 IC50 = 670 nM T80975 C75NGL 44384514 IC50 = 1100 nM T80975 CI2L9R 44384964 IC50 > 1000 nM T80975 CQGW07 44385080 IC50 = 1000 nM T80975 CL4Y9M 44385116 IC50 > 1000 nM T80975 C8EIN0 44387663 IC50 > 10000 nM T80975 CX6YU4 44388576 IC50 = 55 nM T80975 C1NRD0 44389710 IC50 = 18 nM T80975 CH65PU 44389753 IC50 = 7 nM T80975 CCB1X5 44389793 IC50 = 64 nM T80975 C93BDT 44389809 IC50 = 55 nM T80975 C3M6FW 44389820 IC50 = 14 nM T80975 CFD5W4 44389826 IC50 = 190 nM T80975 CZM47F 44389835 IC50 = 380 nM T80975 C5IVA4 44389838 IC50 = 310 nM T80975 C1AJC9 44389849 IC50 = 370 nM T80975 CC2D5H 44389860 IC50 = 33 nM T80975 CELA64 44389975 IC50 = 5 nM T80975 C8ID4C 44389982 IC50 = 4 nM T80975 C3H4OJ 44389991 IC50 = 5 nM T80975 C2J5IU 44395427 IC50 = 410 nM T80975 CV8XB0 44395460 IC50 = 140 nM T80975 CKWY10 44395496 IC50 = 160 nM T80975 C5WYF8 44395528 IC50 = 470 nM T80975 CKT92S 44395562 IC50 = 720 nM T80975 CSBC59 44396134 IC50 > 20000 nM T80975 CW3BP8 44398371 IC50 = 510 nM T80975 CWR4Q0 44398656 IC50 = 180 nM T80975 CUA37S 44398657 IC50 = 96 nM T80975 CZ7TN1 44398732 IC50 = 180 nM T80975 CA5M3C 44400503 IC50 = 65 nM T80975 CR1D2K 44402861 IC50 = 1200 nM T80975 C8QW4A 44402862 IC50 = 1300 nM T80975 CT8IQ7 44402863 IC50 = 100 nM T80975 C8A4JK 44402864 IC50 = 400 nM T80975 C5NE9Y 44402865 IC50 = 4100 nM T80975 CW23JS 44402866 IC50 = 130 nM T80975 C6PFJ1 44402867 IC50 = 3100 nM T80975 CRD24A 44405548 IC50 = 5500 nM T80975 CD2T6B 44405551 IC50 = 30 nM T80975 COSI79 44405552 IC50 = 30 nM T80975 C5E0NF 44405556 IC50 = 80 nM T80975 C2M7EK 44405584 IC50 = 570 nM T80975 CK84OX 44405585 IC50 = 2700 nM T80975 CQ95VK 44405700 IC50 = 3600 nM T80975 C4ZN5K 44405706 IC50 = 680 nM T80975 C3NKD4 44405727 IC50 < 2 nM T80975 C1IZU5 44405750 IC50 = 1900 nM T80975 C68GPB 44405755 IC50 = 2900 nM T80975 CYS5N9 44405756 IC50 = 900 nM T80975 CGI5L7 44405938 IC50 = 16000 nM T80975 C0G3WF 44405939 IC50 > 20000 nM T80975 CR3Q7Z 44405940 IC50 > 20000 nM T80975 C79WRL 44405941 IC50 = 12000 nM T80975 C9ZNA0 44405945 IC50 > 100000 nM T80975 C9LD2T 44405946 IC50 > 100000 nM T80975 C0RO6U 44405949 IC50 = 20000 nM T80975 CC67EN 44405964 IC50 < 1000 nM T80975 C2CTN7 44405982 IC50 = 23000 nM T80975 C0CR1O 44405983 IC50 > 100000 nM T80975 CW86VI 44405987 IC50 > 100000 nM T80975 C5V4TQ 44405999 IC50 = 8000 nM T80975 C0XZ8K 44406013 IC50 = 2000 nM T80975 CS3K1P 44406014 IC50 = 510 nM T80975 CC93JP 44406018 IC50 = 4000 nM T80975 C7P0IH 44406019 IC50 = 19000 nM T80975 CAVE92 44406020 IC50 = 4800 nM T80975 CJW6L4 44406041 IC50 = 1500 nM T80975 C4X2ME 44406047 IC50 = 17000 nM T80975 C36YDV 44406048 IC50 = 11000 nM T80975 CTPE63 44406049 IC50 < 1000 nM T80975 CXZ5C3 44406055 IC50 = 6000 nM T80975 CCRZ12 44406074 IC50 = 490 nM T80975 CUA18B 44407238 IC50 = 13000 nM T80975 CR3O1C 44407275 IC50 = 12600 nM T80975 C70BFV 44407276 IC50 = 15500 nM T80975 CMH7W6 44407277 IC50 = 5500 nM T80975 C7RUK0 44407326 IC50 = 62 nM T80975 CUZ3R7 44407428 IC50 = 600 nM T80975 CIJ21W 44407451 IC50 = 2500 nM T80975 CDR8H1 44408191 IC50 = 2600 nM T80975 CWB0S4 44408195 IC50 > 10000 nM T80975 C4QYG3 44408198 IC50 > 10000 nM T80975 CXG0P1 44408202 IC50 > 10000 nM T80975 COY37U 44408215 IC50 = 170 nM T80975 C4Q6AU 44408662 IC50 = 46 nM T80975 CQS1C8 44408663 IC50 = 710 nM T80975 CO9Y5V 44408666 IC50 = 64 nM T80975 CMK9U8 44408667 IC50 > 10000 nM T80975 CE69KV 44408690 IC50 > 10000 nM T80975 CZ7EC3 44408694 IC50 = 180 nM T80975 CG8FQ3 44408695 IC50 = 52 nM T80975 COKT15 44408845 IC50 > 10000 nM T80975 C0UZB8 44408850 IC50 = 3540 nM T80975 CJC51Y 44408863 IC50 = 1050 nM T80975 CKT3D9 44408868 IC50 = 440 nM T80975 CZU6Y2 44408869 IC50 = 130 nM T80975 C6E9XY 44408879 IC50 = 43 nM T80975 CH2V8K 44408916 IC50 = 66 nM T80975 CHZ7R4 44408923 IC50 = 640 nM T80975 C6DKJ9 44408924 IC50 = 140 nM T80975 CB71IO 44408930 IC50 = 730 nM T80975 C04IOD 44408931 IC50 = 3220 nM T80975 CIQ75Y 44408972 IC50 > 10000 nM T80975 CR4X5E 44408975 IC50 > 10000 nM T80975 C5VN0R 44409048 IC50 > 10000 nM T80975 CJE32H 44409051 IC50 = 280 nM T80975 CSZ9Y5 44409052 IC50 = 210 nM T80975 CZJP10 44409058 IC50 = 66 nM T80975 CC9NV5 44409070 IC50 > 10000 nM T80975 CNT4R5 44409071 IC50 = 3550 nM T80975 CT4O5I 44409087 IC50 = 470 nM T80975 CJIC91 44409090 IC50 = 350 nM T80975 C0C5FS 44409091 IC50 > 10000 nM T80975 CD3Q8H 44409100 IC50 > 10000 nM T80975 C0I3RA 44409105 IC50 = 430 nM T80975 C4WDI5 44409106 IC50 = 92 nM T80975 C6QA8U 44409110 IC50 = 230 nM T80975 CFZ05Y 44409111 IC50 > 10000 nM T80975 CKJ8I0 44409136 IC50 = 110 nM T80975 CST12L 44409141 IC50 = 120 nM T80975 CI71ZK 44409142 IC50 = 4280 nM T80975 CBX37N 44409151 IC50 = 440 nM T80975 C2M8WP 44409154 IC50 = 380 nM T80975 C4JH7R 44409166 IC50 = 690 nM T80975 CRW9G6 44409167 IC50 = 1550 nM T80975 C3Z9HC 44409172 IC50 = 2120 nM T80975 CC5U3T 44409175 IC50 = 5650 nM T80975 CF75LM 44409176 IC50 = 2370 nM T80975 CND3M2 44409185 IC50 = 2000 nM T80975 C6E9ZO 44409186 IC50 > 10000 nM T80975 C5S6UA 44409188 IC50 > 10000 nM T80975 C26DKP 44409192 IC50 = 52 nM T80975 CRN61C 44409200 IC50 = 250 nM T80975 C1E9AZ 44409202 IC50 > 10000 nM T80975 CY80ID 44409203 IC50 > 10000 nM T80975 C2ZAL9 44409207 IC50 = 960 nM T80975 CKM2X3 44409224 IC50 = 95 nM T80975 C72OPJ 44409254 IC50 > 10000 nM T80975 CX0DN5 44409262 IC50 = 61 nM T80975 C05SDW 44409266 IC50 = 87 nM T80975 C21FOV 44409267 IC50 = 110 nM T80975 CUK1I5 44409271 IC50 = 73 nM T80975 C16QCJ 44409285 IC50 = 56 nM T80975 C1W7AS 44409294 IC50 = 310 nM T80975 CJ15KO 44409300 IC50 = 2660 nM T80975 CC79ES 44409305 IC50 > 10000 nM T80975 CH15MA 44409306 IC50 > 10000 nM T80975 C29AMO 44409313 IC50 > 10000 nM T80975 CGO3A8 44409320 IC50 = 440 nM T80975 CBM5T2 44409324 IC50 = 290 nM T80975 C8WJ1O 44409325 IC50 = 210 nM T80975 C5SH2J 44409329 IC50 = 130 nM T80975 CO0ZG9 44409334 IC50 = 75 nM T80975 CAZ70W 44409374 IC50 = 390 nM T80975 CMGA85 44409431 IC50 = 230 nM T80975 C1M4OG 44409433 IC50 = 79 nM T80975 CF7N4T 44409559 IC50 = 210 nM T80975 C9RY1D 44409569 IC50 = 87 nM T80975 CQ90DO 44409594 IC50 = 310 nM T80975 C1OAD0 44409595 IC50 = 470 nM T80975 C8T5UC 44409596 IC50 = 78 nM T80975 CP4C2F 44410079 IC50 = 17 nM T80975 CB26QC 44410112 IC50 = 59 nM T80975 CYNW20 44410113 IC50 = 45 nM T80975 C1MJD7 44410204 IC50 = 23 nM T80975 C6BMZ3 44410265 IC50 = 10 nM T80975 C8MI6F 44410266 IC50 = 30 nM T80975 C0Q5KU 44410267 IC50 = 17 nM T80975 CTSA39 44410333 IC50 = 6 nM T80975 CLF0J2 44410334 IC50 = 26 nM T80975 CV09DY 44410717 IC50 > 10000 nM T80975 CP3CI1 44410720 IC50 > 10000 nM T80975 C8W7AD 44410723 IC50 > 10000 nM T80975 CAT5X4 44410829 IC50 > 10000 nM T80975 CC6Y5P 44410844 IC50 > 10000 nM T80975 CG34TY 44410851 IC50 > 10000 nM T80975 C41EIA 44410869 IC50 > 10000 nM T80975 CB6AE8 44410948 IC50 > 10000 nM T80975 CXZG12 44410949 IC50 > 10000 nM T80975 CS7IE9 44410953 IC50 > 10000 nM T80975 CA9M4X 44410954 IC50 > 10000 nM T80975 C3SP5H 44410955 IC50 > 10000 nM T80975 C5D6YP 44410956 IC50 > 10000 nM T80975 C5W1VC 44410959 IC50 > 10000 nM T80975 CM1C2G 44410960 IC50 > 10000 nM T80975 CVSI80 44411048 IC50 > 10000 nM T80975 CN72BR 44411161 IC50 > 10000 nM T80975 C4AW0O 44411183 IC50 > 10000 nM T80975 C26AZB 44414307 IC50 = 2777 nM T80975 CS8YQ2 44414316 IC50 = 18 nM T80975 C7KZV2 44414322 IC50 = 147 nM T80975 CFM39X 44414323 IC50 = 212 nM T80975 CJM06T 44414347 IC50 = 180 nM T80975 CBZ2X3 44414348 IC50 = 48 nM T80975 C84DVH 44414371 IC50 = 180 nM T80975 C32UEI 44414376 IC50 = 61 nM T80975 C45PBG 44414394 IC50 = 45 nM T80975 CD1I5Y 44414395 IC50 = 171 nM T80975 CG0XV6 44414401 IC50 = 180 nM T80975 CF2JA5 44414419 IC50 = 198 nM T80975 CFGE73 44414421 IC50 = 102 nM T80975 C3G2FJ 44414460 IC50 = 184 nM T80975 C6YL5H 44414486 IC50 = 159 nM T80975 C5RTK0 44414527 IC50 = 19 nM T80975 CRL1C4 44414547 IC50 = 164 nM T80975 C0MZ7P 44414549 IC50 = 21 nM T80975 C3SYD7 44414595 IC50 = 123 nM T80975 CP6TZ2 44414596 IC50 = 262 nM T80975 C6I8TW 44414597 IC50 = 17 nM T80975 CIQA35 44414621 IC50 = 21 nM T80975 CUW8C1 44414632 IC50 = 259 nM T80975 C06UCM 44414633 IC50 = 12 nM T80975 C2PK5Z 44414637 IC50 = 12285 nM T80975 CQB17H 44414646 IC50 = 20 nM T80975 CLD07U 44414647 IC50 = 27 nM T80975 CTAZ73 44414648 IC50 = 16 nM T80975 CK9OQ7 44414658 IC50 > 50000 nM T80975 C1XCW7 44414659 IC50 = 199 nM T80975 C2WE7V 44414665 IC50 = 459 nM T80975 C1TR2Y 44414666 IC50 = 63 nM T80975 CBY7D9 44414679 IC50 = 4 nM T80975 C8HJ9Z 44414682 IC50 = 22795 nM T80975 CO14UX 44414683 IC50 = 444 nM T80975 C7Q0ID 44414688 IC50 = 8600 nM T80975 CKU21Y 44414689 IC50 = 2100 nM T80975 C5KML9 44414694 IC50 > 50000 nM T80975 C1LZ9S 44414695 IC50 = 308 nM T80975 C1J4YF 44414702 IC50 = 22000 nM T80975 CI4H6L 44414703 IC50 = 16000 nM T80975 CK7EZ4 44414706 IC50 = 24158 nM T80975 CS5JX0 44414742 IC50 > 50000 nM T80975 CIU45K 44414743 IC50 = 46000 nM T80975 CBDR90 44414759 IC50 = 43000 nM T80975 C6DH0Q 44414776 IC50 > 50000 nM T80975 C0JF1Z 44414779 IC50 = 16 nM T80975 C0THE4 44414816 IC50 = 79 nM T80975 C1DSL3 44414828 IC50 = 5 nM T80975 CFV84D 44414841 IC50 = 19 nM T80975 CRF01G 44414847 IC50 = 2882 nM T80975 CXV94N 44414848 IC50 = 4807 nM T80975 C19SVU 44414855 IC50 = 14100 nM T80975 C8PBJ1 44414866 IC50 = 42 nM T80975 CUI2N3 44414867 IC50 = 34 nM T80975 C8LH5Q 44414868 IC50 = 7458 nM T80975 CG72ML 44414871 IC50 = 708 nM T80975 C5AFO9 44414872 IC50 = 600 nM T80975 CICB10 44414879 IC50 > 50000 nM T80975 CD13BL 44414880 IC50 = 281 nM T80975 CTCM71 44414881 IC50 = 122 nM T80975 C89MTI 44414963 IC50 = 2840 nM T80975 C75WHY 44414964 IC50 = 143000 nM T80975 C2P0UL 44414965 IC50 = 824000 nM T80975 C5FN3S 44414971 IC50 = 7480 nM T80975 CGTX67 44414972 IC50 = 16640 nM T80975 CU7G2Q 44414973 IC50 = 190000 nM T80975 C9QAG6 44414974 IC50 = 4081000 nM T80975 CI8B5H 44414979 IC50 = 5470 nM T80975 C0FW2L 44414980 IC50 = 12540 nM T80975 CCBK18 44414981 IC50 = 665000 nM T80975 CW7G6C 44414982 IC50 = 190000 nM T80975 CO8U5B 44414993 IC50 = 1050 nM T80975 C5L2TP 44414994 IC50 > 50000 nM T80975 C4U1IA 44414995 IC50 > 50000 nM T80975 CI36HR 44414996 IC50 = 108000 nM T80975 C9V7LN 44415005 IC50 = 3400 nM T80975 CC31TM 44415007 IC50 = 400 nM T80975 CI4SH2 44415008 IC50 = 1005000 nM T80975 C3FCG6 44415015 IC50 = 9200 nM T80975 C8G5YN 44415111 IC50 = 350 nM T80975 CHJ7T1 44415158 IC50 = 200 nM T80975 C5TQ4F 44415291 IC50 = 570 nM T80975 C5R7IW 44416429 IC50 > 10000 nM T80975 C7C4TK 44416433 IC50 > 10000 nM T80975 C0IUL9 44416434 IC50 > 10000 nM T80975 CR42NY 44416467 IC50 > 10000 nM T80975 C41SAP 44416508 IC50 > 10000 nM T80975 CK8R2O 44416545 IC50 > 10000 nM T80975 CX17JM 44416560 IC50 = 2000 nM T80975 CD2FC0 44416568 IC50 > 10000 nM T80975 CPIA51 44416569 IC50 > 10000 nM T80975 CX3DU9 44416596 IC50 > 10000 nM T80975 C35BCH 44416635 IC50 > 10000 nM T80975 C6HQ5D 44416655 IC50 > 10000 nM T80975 CIV18H 44416687 IC50 = 2000 nM T80975 C43VZI 44416688 IC50 = 2000 nM T80975 CF5UH3 44416692 IC50 > 10000 nM T80975 C43NYR 44416693 IC50 > 10000 nM T80975 C8RHO3 44416712 IC50 = 2000 nM T80975 CZ3WQ2 44416741 IC50 > 10000 nM T80975 CLQ8W9 44417523 IC50 > 5000 nM T80975 C2LDT6 44417577 IC50 > 33000 nM T80975 C7F8GP 44417581 IC50 = 21500 nM T80975 C7HQ1V 44418298 IC50 = 11 nM T80975 CO9H4N 44418299 IC50 = 11 nM T80975 CJF6B1 44418302 IC50 = 16 nM T80975 CYP61S 44418305 IC50 = 14 nM T80975 C6YW3N 44418309 IC50 = 8 nM T80975 C9W3GM 44418314 IC50 = 21 nM T80975 C3VD2Z 44418318 IC50 = 29 nM T80975 CT3N1H 44418321 IC50 = 16 nM T80975 CT12WM 44418327 IC50 = 7 nM T80975 C7J2XU 44418332 IC50 = 12 nM T80975 C7IO3E 44418339 IC50 = 12 nM T80975 CS25UA 44418346 IC50 = 9 nM T80975 CG49MW 44418350 IC50 = 48 nM T80975 CB1W8D 44418356 IC50 = 9 nM T80975 CN74KG 44418361 IC50 = 18 nM T80975 CAC8R3 44418362 IC50 = 101 nM T80975 C6W1LF 44418363 IC50 = 24 nM T80975 C01OZP 44418364 IC50 = 159 nM T80975 CM7OV4 44418365 IC50 = 25 nM T80975 CY8UZ5 44418366 IC50 = 41 nM T80975 CM9YH8 44418374 IC50 = 9 nM T80975 CZW1V5 44418379 IC50 = 3 nM T80975 C1DLQ9 44418386 IC50 = 5 nM T80975 C0NF4E 44418392 IC50 = 12 nM T80975 CVP5Q4 44418397 IC50 = 46 nM T80975 CT6ZD3 44418402 IC50 = 2 nM T80975 CLIY92 44418410 IC50 = 3 nM T80975 CFEA89 44418422 IC50 = 88 nM T80975 CLO5F6 44418448 IC50 = 10 nM T80975 CG5FS7 44418453 IC50 = 4 nM T80975 C1YGN9 44418460 IC50 = 7 nM T80975 C89MBJ 44418993 IC50 = 2600 nM T80975 C31XOY 44418994 IC50 > 25000 nM T80975 C16KGX 44420777 IC50 = 13 nM T80975 C51BYS 44420784 IC50 = 86 nM T80975 C0K1JL 44420785 IC50 = 21 nM T80975 CZ8CW6 44420786 IC50 = 15 nM T80975 CXZ2L3 44421702 IC50 = 9 nM T80975 CT0J7Z 44421703 IC50 = 1000 nM T80975 C5WGQ0 44421704 IC50 = 146 nM T80975 CF34KY 44421705 IC50 = 51 nM T80975 C4OF6A 44425581 IC50 > 12500 nM T80975 C9X2NC 44425583 IC50 = 25 nM T80975 CO7X8F 44425786 IC50 = 4 nM T80975 C3QJF6 44425788 IC50 = 30 nM T80975 C3MPT1 44425791 IC50 = 90 nM T80975 CWBD93 44425808 IC50 = 13 nM T80975 C95AYW 44425813 IC50 = 60 nM T80975 CKI50A 44425816 IC50 = 380 nM T80975 CETQ79 44427518 IC50 > 50000 nM T80975 COPG94 44427519 IC50 > 10000 nM T80975 C1U4JB 44427900 Ki = 1.6 nM T80975 CRP04Z 44428103 IC50 = 510 nM T80975 C0PLD7 44428887 IC50 = 109.3 nM T80975 C2V1FP 44428888 IC50 = 113.4 nM T80975 C2UT9G 44428889 IC50 = 550.2 nM T80975 C8XRO1 44428890 IC50 = 783.1 nM T80975 C3A2HC 44428891 IC50 = 135 nM T80975 C42KHG 44428893 IC50 = 80.2 nM T80975 CDE73U 44428895 IC50 = 76.2 nM T80975 C5H3DV 44428898 IC50 = 371.5 nM T80975 C2V1ER 44428899 IC50 = 188.7 nM T80975 CLGZ52 44428901 IC50 = 4389 nM T80975 C8LI7S 44428906 IC50 = 50.2 nM T80975 C2U5KW 44430873 IC50 = 61 nM T80975 C0P8BA 44430874 IC50 = 91 nM T80975 CQXL12 44430875 IC50 = 110 nM T80975 C25WQT 44430876 IC50 = 180 nM T80975 C9I2GJ 44430877 IC50 = 360 nM T80975 CKCX40 44430878 IC50 = 380 nM T80975 C0ZXY6 44430879 IC50 = 410 nM T80975 CL7C6R 44430880 IC50 = 490 nM T80975 CS9O6C 44430882 IC50 = 2100 nM T80975 C98QBK 44430883 IC50 = 10000 nM T80975 CD8B4J 44430884 IC50 > 10000 nM T80975 C7PNC9 44430885 IC50 > 10000 nM T80975 CY6P9J 44430886 IC50 > 10000 nM T80975 C8MLH2 44430887 IC50 > 10000 nM T80975 CNU34S 44430906 IC50 = 52 nM T80975 CLEX18 44430913 IC50 = 90 nM T80975 CZIC28 44430916 IC50 = 150 nM T80975 C2J5XB 44430917 IC50 = 180 nM T80975 CBQM21 44430920 IC50 = 200 nM T80975 CQ7L8Y 44430921 IC50 = 340 nM T80975 CDW6L0 44430924 IC50 = 410 nM T80975 CXK2J8 44430925 IC50 = 1400 nM T80975 CA0N4B 44430927 IC50 = 1600 nM T80975 CQN31M 44430929 IC50 = 21 nM T80975 CL7X4E 44430931 IC50 = 450 nM T80975 CG4E1T 44431447 IC50 = 348 nM T80975 C5QWY4 44431448 IC50 = 33 nM T80975 CP76WK 44431449 IC50 = 19 nM T80975 CR1G5K 44431450 IC50 = 159 nM T80975 CJ64DM 44431451 IC50 = 797 nM T80975 C0XFS5 44431452 IC50 = 7 nM T80975 C5VPN4 44431453 IC50 = 216 nM T80975 CE81LF 44431454 IC50 = 103 nM T80975 CGK6T3 44431455 IC50 = 15 nM T80975 C0NZX8 44431456 IC50 = 455 nM T80975 CE7N4S 44431457 IC50 = 314 nM T80975 C4R6AN 44431460 IC50 = 7 nM T80975 CJM89C 44431461 IC50 = 37 nM T80975 CND24H 44431888 IC50 > 10000 nM T80975 CJHD30 44431889 IC50 > 10000 nM T80975 C5X8IO 44431890 IC50 = 77 nM T80975 CF31BX 44431891 IC50 > 10000 nM T80975 C6DME5 44431892 IC50 > 10000 nM T80975 CK1AS2 44431893 IC50 > 10000 nM T80975 CJ73EF 44431894 IC50 > 10000 nM T80975 C3SG5E 44431895 IC50 > 10000 nM T80975 C6VZ8W 44431896 IC50 > 10000 nM T80975 C6YL7I 44431897 IC50 = 48 nM T80975 CU4MN1 44431898 IC50 = 86 nM T80975 CTR14P 44431899 IC50 = 18 nM T80975 C8OWB5 44431900 IC50 = 280 nM T80975 C2IJ4Q 44431901 IC50 = 21 nM T80975 C2Y4XS 44431902 IC50 = 42 nM T80975 CME54X 44431903 IC50 = 53 nM T80975 C0KM8Y 44431904 IC50 = 950 nM T80975 C5B2EM 44431905 IC50 = 3220 nM T80975 C79PXH 44431906 IC50 > 10000 nM T80975 CRC6N1 44431907 IC50 = 180 nM T80975 C46YKU 44431908 IC50 = 5150 nM T80975 CJSK07 44431909 IC50 > 10000 nM T80975 C36QDE 44431910 IC50 = 450 nM T80975 CET6B3 44431911 IC50 = 95 nM T80975 CUM12J 44431912 IC50 = 260 nM T80975 CB73ES 44431913 IC50 = 90 nM T80975 C35AGI 44431914 IC50 = 780 nM T80975 C75NGZ 44431915 IC50 = 1190 nM T80975 C6ANT8 44431916 IC50 > 10000 nM T80975 CD4QB5 44431917 IC50 > 10000 nM T80975 CPRX24 44431918 IC50 > 10000 nM T80975 CL85AI 44431919 IC50 > 10000 nM T80975 CP68DH 44431920 IC50 = 380 nM T80975 CDX70N 44431921 IC50 = 470 nM T80975 CXQ4K6 44431922 IC50 = 1050 nM T80975 C8Q1XM 44431925 IC50 = 940 nM T80975 C9NY4F 44431927 IC50 = 4950 nM T80975 C6C5GM 44431928 IC50 > 10000 nM T80975 CTL31N 44431930 IC50 > 10000 nM T80975 C58POW 44431932 IC50 > 10000 nM T80975 CZT4Y3 44431935 IC50 = 640 nM T80975 C1O5QH 44431936 IC50 = 2960 nM T80975 CGR4F6 44431939 IC50 = 2650 nM T80975 C6EL0U 44431940 IC50 > 10000 nM T80975 C1Z6NQ 44431941 IC50 > 10000 nM T80975 CF72BI 44432051 IC50 > 10000 nM T80975 CQWC12 44438817 IC50 = 30 nM T80975 C0YU5D 44439355 IC50 > 10000 nM T80975 C4UO8C 44439356 IC50 = 3120 nM T80975 C0IXS5 44439357 IC50 = 2550 nM T80975 CL7Q0Z 44439358 IC50 > 10000 nM T80975 CGSR93 44439359 IC50 = 550 nM T80975 CT3B4P 44439360 IC50 = 6000 nM T80975 CWS7D3 44439361 IC50 = 110 nM T80975 COYR48 44439362 IC50 = 350 nM T80975 C1PIW8 44439363 IC50 = 1650 nM T80975 CZP54X 44439364 IC50 = 3220 nM T80975 C1CB7D 44439365 IC50 = 75 nM T80975 C3QH1P 44439366 IC50 > 10000 nM T80975 C9GH4W 44439367 IC50 > 10000 nM T80975 CLME26 44439368 IC50 > 10000 nM T80975 C1S3IP 44439369 IC50 = 350 nM T80975 C5YT3N 44439448 IC50 > 10000 nM T80975 CK1O5J 44439449 IC50 = 170 nM T80975 C9XE4V 44439450 IC50 = 88 nM T80975 C75DRT 44439451 IC50 = 96 nM T80975 CXI3B5 44439452 IC50 = 57 nM T80975 CZ5T6X 44439453 IC50 = 110 nM T80975 C4C0XH 44439454 IC50 = 150 nM T80975 C37IHP 44439455 IC50 = 89 nM T80975 C13TLQ 44439457 Ki = 0.16 nM T80975 CZM4Y0 44439458 IC50 = 1350 nM T80975 CO29LB 44439459 IC50 = 740 nM T80975 CY76DC 44439460 IC50 > 10000 nM T80975 C35RTN 44439461 IC50 > 10000 nM T80975 CU2SG9 44439462 IC50 > 10000 nM T80975 CG0A7Z 44439463 IC50 > 10000 nM T80975 C4R8HQ 44439464 IC50 = 1060 nM T80975 CDQ6K8 44439465 IC50 = 130 nM T80975 C6DQV9 44439466 Ki = 0.17 nM T80975 CVP1S9 44439467 IC50 = 470 nM T80975 C5VL4O 44439468 IC50 = 1000 nM T80975 CS49IA 44439469 IC50 = 3220 nM T80975 CN65DW 44439470 IC50 = 45 nM T80975 C4BJI2 44439471 IC50 = 88 nM T80975 CTU07B 44439472 IC50 > 10000 nM T80975 C1WFV5 44439475 IC50 > 10000 nM T80975 CE1U3I 44439478 IC50 > 10000 nM T80975 CBC3V5 44439479 IC50 = 520 nM T80975 CQ9Y7K 44439480 IC50 = 110 nM T80975 C97RIN 44439481 IC50 = 79 nM T80975 CI75KD 44439482 IC50 = 82 nM T80975 C03YPU 44439484 IC50 = 91 nM T80975 CL7KY8 44439487 IC50 = 130 nM T80975 CYU6S0 44439495 IC50 = 210 nM T80975 C05LUV 44439496 IC50 = 930 nM T80975 C9J0IC 44439497 IC50 = 69 nM T80975 C6A3OB 44439499 IC50 = 2270 nM T80975 CH6FM2 44439501 IC50 = 180 nM T80975 C09HPL 44439502 IC50 = 910 nM T80975 C98OAT 44439503 IC50 > 10000 nM T80975 CA81EQ 44439504 IC50 > 10000 nM T80975 CLFS52 44439505 IC50 > 10000 nM T80975 C8YZ0F 44439506 IC50 = 210 nM T80975 C9M4SR 44439507 IC50 = 350 nM T80975 C09PNG 44439508 IC50 > 10000 nM T80975 C7F1SN 44439509 IC50 > 10000 nM T80975 C25SEZ 44439510 IC50 > 10000 nM T80975 CR5K0Q 44439511 IC50 = 1220 nM T80975 CQ0E2J 44439512 IC50 > 10000 nM T80975 COC5E7 44439513 IC50 = 320 nM T80975 CQO50A 44439514 IC50 = 930 nM T80975 C9KC5D 44439515 IC50 = 3350 nM T80975 CJL03B 44439516 IC50 > 10000 nM T80975 CU4O8W 44439517 IC50 = 590 nM T80975 C14MTJ 44440231 IC50 = 7040 nM T80975 CA86YP 44440232 IC50 = 4840 nM T80975 COK21X 44440233 IC50 = 27890 nM T80975 CYMN10 44440242 IC50 = 580 nM T80975 C96ARW 44440243 IC50 = 410 nM T80975 CGL0R4 44440244 IC50 = 440 nM T80975 CQI8S3 44440245 IC50 = 560 nM T80975 CZM08I 44440246 IC50 = 70 nM T80975 C4O8NF 44440247 IC50 = 650 nM T80975 C1DAU0 44440248 IC50 = 310 nM T80975 C93TBM 44440249 IC50 = 50 nM T80975 C6VLC0 44440250 IC50 = 110 nM T80975 CO37FE 44440251 IC50 = 60 nM T80975 C6T0IK 44440252 IC50 = 100 nM T80975 CJ05OC 44440253 IC50 = 920 nM T80975 CGV37F 44440254 IC50 = 53 nM T80975 C5JUV3 44440256 IC50 = 270 nM T80975 CFB56S 44440259 IC50 = 36 nM T80975 CEW9G2 44440261 IC50 = 263 nM T80975 CL52XP 44440291 IC50 = 38 nM T80975 CQX84Z 44440292 IC50 = 20 nM T80975 C35NRO 44440293 IC50 = 5 nM T80975 CZE89H 44440294 IC50 = 2 nM T80975 C2UG3R 44440295 IC50 = 117 nM T80975 CXD5L8 44440296 IC50 = 18 nM T80975 CK5UH6 44440297 IC50 = 456 nM T80975 CSBX36 44440298 IC50 = 128 nM T80975 CD81OT 44440299 IC50 = 25000 nM T80975 C1HRG0 44440300 IC50 = 18 nM T80975 C1KN2U 44440301 IC50 = 9 nM T80975 CBH1R5 44440302 IC50 = 309 nM T80975 CPB2Z6 44440303 IC50 = 442 nM T80975 C6RC4L 44440304 IC50 = 1126 nM T80975 CGN1Q4 44440305 IC50 = 233 nM T80975 CHP41T 44442415 IC50 = 43 nM T80975 CI26UX 44442416 IC50 = 62 nM T80975 C2W1RN 44442417 IC50 = 7 nM T80975 C4A9FD 44442418 IC50 = 3 nM T80975 C5R4QE 44442729 Ki = 2100 nM T80975 CGC76I 44442730 Ki > 10000 nM T80975 CJM6N5 44442731 Ki > 10000 nM T80975 CH2FS6 44442732 Ki = 2600 nM T80975 CZ7FC6 44442733 Ki = 150 nM T80975 C6PNZ4 44442734 Ki = 560 nM T80975 C8N1EQ 44442735 Ki = 650 nM T80975 C26EVP 44442736 Ki = 99 nM T80975 C0S6PN 44442737 Ki = 140 nM T80975 CAZ5O7 44442738 Ki = 420 nM T80975 CM9XW1 44442739 Ki > 10000 nM T80975 CFOH51 44442740 Ki > 10000 nM T80975 CX10DZ 44442742 Ki = 1500 nM T80975 CN12IA 44442744 Ki > 10000 nM T80975 C0DOP6 44442745 Ki = 170 nM T80975 C6LW5U 44443795 Ki = 140 nM T80975 CC4K1I 44443796 Ki > 10000 nM T80975 C6J7MT 44443810 Ki = 29 nM T80975 CE6I5G 44443811 Ki > 6660 nM T80975 CD7NH9 44443815 Ki = 135 nM T80975 CA9R0H 44443817 Ki > 20000 nM T80975 C1L6MG 44444041 IC50 = 530 nM T80975 CWI4H7 44446962 IC50 = 380 nM T80975 CG5FA3 44447873 IC50 = 3 nM T80975 CM6A1T 44447874 IC50 = 18 nM T80975 CJ6T9P 44447875 IC50 = 4 nM T80975 CD20WZ 44447876 IC50 = 1 nM T80975 CPY39Q 44447877 IC50 = 2 nM T80975 C4JD3N 44447878 IC50 = 4 nM T80975 C2K6ZS 44447879 IC50 = 23 nM T80975 C2NMO0 44447881 IC50 = 3 nM T80975 CB2N8J 44447882 IC50 = 4 nM T80975 CSF9U6 44447883 IC50 = 31 nM T80975 C2BP9I 44447884 IC50 = 5 nM T80975 C9MPX0 44447885 IC50 = 4 nM T80975 C1M0DP 44447887 IC50 = 1 nM T80975 CTXY59 44447888 IC50 = 4 nM T80975 C4YMI9 44447890 IC50 = 4 nM T80975 C7L9AF 44447891 IC50 = 12 nM T80975 CHR96X 44447892 IC50 = 4 nM T80975 CZ8DG5 44447893 IC50 = 4 nM T80975 C5X2HE 44447894 IC50 = 94 nM T80975 CR65PM 44447895 IC50 = 4 nM T80975 CQH8F7 44447896 IC50 = 4 nM T80975 C3PH2E 44447897 IC50 = 2 nM T80975 CSB53H 44447898 IC50 = 3 nM T80975 CZJ3B9 44449300 IC50 > 1000 nM T80975 C61KOC 44449479 IC50 = 25 nM T80975 CU4A9F 44449484 IC50 = 150 nM T80975 C8GT4I 44449507 IC50 = 36 nM T80975 CUB12D 44449577 IC50 = 31 nM T80975 CY8G9C 44449578 IC50 = 113 nM T80975 C5X0JD 44449609 IC50 = 96 nM T80975 CC02TP 44449644 IC50 = 17 nM T80975 C69KRH 44449674 IC50 = 121 nM T80975 C6I5WJ 44449677 IC50 = 165 nM T80975 CA5EI1 44449715 IC50 = 223 nM T80975 CX0VR5 44449716 IC50 = 122 nM T80975 C13FIN 44450007 IC50 > 13000 nM T80975 CZ1R8M 44450033 IC50 = 21000 nM T80975 CIY3T5 44450035 IC50 = 600 nM T80975 C5Y4PN 44450059 IC50 = 3000 nM T80975 C28LMV 44450060 IC50 = 4000 nM T80975 C3ZBV8 44450546 IC50 = 70 nM T80975 CXL80U 44453148 IC50 = 75 nM T80975 C06KUB 44453149 IC50 = 21 nM T80975 CGA6S8 44453150 IC50 = 3 nM T80975 CMPZ16 44453151 IC50 = 26 nM T80975 C3DLE8 44453187 IC50 = 10 nM T80975 CC6EP9 44453188 IC50 = 13 nM T80975 CYS5W1 44453216 IC50 = 35 nM T80975 C6E2SG 44453252 IC50 = 17 nM T80975 C6TMR8 44453253 IC50 = 15 nM T80975 C4U7ZB 44453254 IC50 = 16 nM T80975 CQ9Y3M 44453489 IC50 = 10 nM T80975 CDV6X9 44454507 IC50 > 25000 nM T80975 C6SMY7 44454538 IC50 = 8330 nM T80975 C3EAH1 44454630 IC50 = 57 nM T80975 CK4O2M 44454632 IC50 = 200 nM T80975 CZI92T 44454651 IC50 = 6679 nM T80975 CIA39D 44454676 IC50 > 25000 nM T80975 C7DGA2 44454678 IC50 > 25000 nM T80975 C0MF7P 44454684 IC50 = 21 nM T80975 C1F3LT 44454702 IC50 = 2030 nM T80975 CCW57R 44454703 IC50 > 25000 nM T80975 CFS7W2 44454728 IC50 > 25000 nM T80975 CTL43P 44454729 IC50 > 25000 nM T80975 CZC95J 44454731 IC50 > 25000 nM T80975 CC56ZN 44454845 IC50 = 38 nM T80975 C6EL0N 44454848 IC50 = 200 nM T80975 C8F0TR 44455389 IC50 = 1120 nM T80975 CCN4L2 44455555 IC50 = 240 nM T80975 C3YSJ4 44455584 IC50 = 64 nM T80975 C5GF6X 44455585 IC50 = 115 nM T80975 C56WNJ 44455675 IC50 = 4 nM T80975 CW0Q4O 44455758 IC50 = 3.7 nM T80975 C43XKP 44457356 IC50 = 3 nM T80975 C67VXQ 44457503 IC50 = 4 nM T80975 C7N2AQ 44473101 IC50 > 25000 nM T80975 C4MG3F 44473102 IC50 = 300 nM T80975 CA85NJ 44473103 IC50 > 1000 nM T80975 CG8M0E 44511408 IC50 = 3 nM T80975 CCPG93 44511409 IC50 = 2.6 nM T80975 CCJ72O 44511410 IC50 = 3.3 nM T80975 C5R2UA 44511411 IC50 = 1.7 nM T80975 CZRE30 44511412 IC50 = 2.5 nM T80975 CZ3EH7 44511473 IC50 = 2.8 nM T80975 CX2RP9 44511474 IC50 = 3 nM T80975 CIYL41 44511482 IC50 = 19700 nM T80975 CPY54G 44511483 IC50 > 100000 nM T80975 CU1TR3 44511484 IC50 = 11 nM T80975 CLI60D 44511486 IC50 > 100000 nM T80975 C9GJV6 44511541 IC50 = 142 nM T80975 C1N7MF 44511547 IC50 = 7.9 nM T80975 C31GFX 44511607 IC50 = 10.3 nM T80975 C3DXU1 44511608 IC50 = 73 nM T80975 CP5LM7 44511610 IC50 = 400 nM T80975 CX8SI7 44511674 IC50 = 285 nM T80975 CR8XV4 44511675 IC50 = 168 nM T80975 C0AN3V 44511676 IC50 = 759 nM T80975 C4QUJ1 44511677 IC50 = 29 nM T80975 C38XTK 44511678 IC50 = 34 nM T80975 CKH3W0 44511679 IC50 = 10 nM T80975 CYR2T9 44511747 IC50 = 3.4 nM T80975 C2W4PI 44511748 IC50 = 2 nM T80975 CJX4R3 44511749 IC50 = 2 nM T80975 C9JML8 44512430 IC50 = 25 nM T80975 COD69F 44512431 IC50 = 28 nM T80975 CYH6P3 44520205 IC50 = 1180 nM T80975 C4WRN5 44541014 IC50 = 50 nM T80975 C0LY6E 44552561 IC50 = 420 nM T80975 C7KRU3 44552562 IC50 = 350 nM T80975 CYV71I 44555430 IC50 = 9.3 nM T80975 C2DQV1 44560448 IC50 = 5 nM T80975 CTJ0D5 44560449 IC50 = 55 nM T80975 CK72TL 44560450 IC50 = 10 nM T80975 CF16QB 44560451 IC50 = 3530 nM T80975 C0U8DH 44560546 IC50 > 5000 nM T80975 CN3I8C 44560547 IC50 = 470 nM T80975 C0M1FW 44560587 IC50 = 748 nM T80975 C18JQN 44560588 IC50 = 114 nM T80975 C19KFW 44560589 IC50 > 5000 nM T80975 CS8GY1 44560640 IC50 > 25000 nM T80975 C6VF0N 44560641 IC50 > 5000 nM T80975 C4JR8C 44560751 IC50 = 168 nM T80975 C6I1TW 44560803 IC50 = 3 nM T80975 CJ19AU 44560804 IC50 = 8 nM T80975 C4YQ5K 44562290 IC50 = 1700 nM T80975 CG6NL4 44562291 IC50 = 370 nM T80975 C7J1MT 44562292 IC50 = 1110 nM T80975 C4I2KF 44562325 IC50 = 800 nM T80975 C1YU9X 44562369 IC50 = 270 nM T80975 C8RX6B 44562370 IC50 = 230 nM T80975 CH9EA5 44562371 IC50 = 160 nM T80975 C3LZM8 44562372 IC50 = 70 nM T80975 CXE96W 44562393 IC50 = 60 nM T80975 CS71VY 44562394 IC50 = 344 nM T80975 CZN9I3 44562395 IC50 = 8 nM T80975 C70KMJ 44562417 IC50 = 2 nM T80975 CE4W5V 44562418 IC50 = 1 nM T80975 C1A4XG 44562420 IC50 > 10000 nM T80975 C3UV2W 44562431 IC50 > 100000 nM T80975 C03DUS 44562601 IC50 = 8 nM T80975 C3XTA7 44562721 Ki > 25000 nM T80975 C4JRB8 44564129 IC50 > 10000 nM T80975 CE7QT2 44564130 IC50 > 10000 nM T80975 CWF0V5 44564187 IC50 > 400000 ug.mL-1 T80975 C3YU8I 44564188 IC50 > 400000 ug.mL-1 T80975 CL87KN 44564189 IC50 > 400000 ug.mL-1 T80975 CZI65G 44564207 IC50 > 400000 ug.mL-1 T80975 CP7FG1 44564296 IC50 > 10000 nM T80975 CTI4C0 44564574 IC50 = 440 nM T80975 CE3MP5 44564575 IC50 = 930 nM T80975 CFM8P1 44564576 IC50 = 630 nM T80975 C18LQG 44564591 IC50 = 800 nM T80975 C9LZT0 44564592 IC50 = 230 nM T80975 CD2CQ0 44564593 IC50 = 8 nM T80975 CPIR15 44564600 IC50 = 980 nM T80975 CP63RZ 44564651 IC50 > 10000 nM T80975 C5P0EK 44564652 IC50 > 10000 nM T80975 CTF0V2 44564653 IC50 > 10000 nM T80975 C3I0CK 44564664 IC50 = 20 nM T80975 CUSN60 44564665 IC50 = 8 nM T80975 CH7OL6 44564666 IC50 = 26 nM T80975 CU3G5Z 44564667 IC50 = 12 nM T80975 C0N2OH 44564668 IC50 = 8 nM T80975 CPRU17 44564669 IC50 = 880 nM T80975 C0DJ2X 44564670 IC50 = 23 nM T80975 CIVF90 44564688 IC50 > 10000 nM T80975 CH0LV3 44564689 IC50 = 5000 nM T80975 C21HAM 44564690 IC50 > 10000 nM T80975 CPG1H5 44564691 IC50 = 5000 nM T80975 CC7E4K 44564705 IC50 > 10000 nM T80975 C42ZEW 44564706 IC50 = 3600 nM T80975 CNXH83 44564707 IC50 = 12 nM T80975 C1JH3T 44564727 IC50 > 10000 nM T80975 C53MCK 44564747 IC50 = 8800 nM T80975 CDI31F 44564748 IC50 = 8900 nM T80975 CA17NT 44564749 IC50 > 10000 nM T80975 CMIZ20 44564750 IC50 > 10000 nM T80975 CSO9F8 44564751 IC50 > 10000 nM T80975 C5JQF1 44564752 IC50 = 1800 nM T80975 C8ATG9 44564787 IC50 > 10000 nM T80975 CM50GS 44564788 IC50 > 10000 nM T80975 C3Q0DX 44564789 IC50 = 1200 nM T80975 CP40XB 44564790 IC50 > 10000 nM T80975 C35NTB 44564791 IC50 = 10000 nM T80975 CJY83G 44564817 IC50 = 960 nM T80975 CLK98G 44564818 IC50 > 10000 nM T80975 CF2D1K 44564819 IC50 = 9200 nM T80975 C3CQ9K 44564820 IC50 > 10000 nM T80975 CI8V2L 44564821 IC50 > 10000 nM T80975 C9PO7J 44564860 IC50 > 10000 nM T80975 C16FJW 44564861 IC50 > 10000 nM T80975 C8AMX5 44564862 IC50 = 640 nM T80975 CTR59U 44564863 IC50 > 10000 nM T80975 C9EY4C 44564864 IC50 = 600 nM T80975 CG5Z7T 44564910 IC50 = 800 nM T80975 CU9O4C 44564911 IC50 = 1000 nM T80975 CXZ15S 44564954 IC50 > 10000 nM T80975 CZ78WJ 44564955 IC50 > 10000 nM T80975 CJ1X9V 44565013 IC50 = 7500 nM T80975 CN2Q3D 44565014 IC50 = 1900 nM T80975 CM2GN3 44565015 IC50 > 10000 nM T80975 C6RV9I 44565016 IC50 = 870 nM T80975 CTK29Y 44565090 IC50 = 4230 nM T80975 CER4M3 44565091 IC50 > 10000 nM T80975 CB3U0T 44565092 IC50 > 10000 nM T80975 C4ZM1N 44565117 IC50 = 0.035 nM T80975 C1RO5W 44565118 IC50 = 37 nM T80975 C6F0SN 44565141 IC50 > 10000 nM T80975 CXS46L 44565142 IC50 = 270 nM T80975 CI5D3M 44565143 IC50 = 590 nM T80975 CKE2W7 44565144 IC50 = 1220 nM T80975 CJD91Q 44565164 IC50 = 20 nM T80975 C2TX8Y 44565165 IC50 = 10 nM T80975 CP6F5U 44565194 IC50 = 270 nM T80975 C1XHB9 44565195 IC50 = 1630 nM T80975 C7P9CB 44565196 IC50 = 770 nM T80975 CVT9H8 44565197 IC50 = 680 nM T80975 CX06UE 44565221 IC50 = 39 nM T80975 CGM09E 44565222 IC50 = 16 nM T80975 CD5A2Z 44568608 IC50 = 1 nM T80975 C3HW7L 44570553 IC50 = 18000 nM T80975 C17PVE 44570554 IC50 > 30000 nM T80975 CLOY92 44570599 IC50 = 3000 nM T80975 CK06LT 44570600 IC50 > 30000 nM T80975 CV91YE 44572385 IC50 = 9800 nM T80975 C3CB2K 44572429 IC50 = 8600 nM T80975 CM2Q8J 44572430 IC50 = 11000 nM T80975 CAN4B0 44572431 IC50 = 1500 nM T80975 CMAT21 44572489 IC50 = 24000 nM T80975 CU1SY9 44572490 IC50 = 46000 nM T80975 CSD74G 44572491 IC50 = 4400 nM T80975 CA9WO3 44572537 IC50 = 9000 nM T80975 C06SLW 44572538 IC50 = 12000 nM T80975 CY8TG3 44572539 IC50 = 4800 nM T80975 C1JR4C 44572540 IC50 = 43000 nM T80975 CZ0PA9 44572581 IC50 = 14000 nM T80975 CD9VR5 44572582 IC50 = 8700 nM T80975 CG5UK0 44572584 IC50 = 8600 nM T80975 CMX32U 44572633 IC50 = 6700 nM T80975 C0N4ZA 44577698 IC50 = 870 nM T80975 C9VXH3 44577699 IC50 > 10000 nM T80975 C4BFY1 44577740 IC50 = 120 nM T80975 C4Q3YF 44577741 IC50 = 74 nM T80975 C5A4ZP 44577742 IC50 = 10000 nM T80975 C6SWF4 44577743 IC50 > 10000 nM T80975 C5XY0R 44577763 IC50 = 2600 nM T80975 C7KF8U 44577764 IC50 = 3000 nM T80975 C9LKX2 44577765 IC50 = 8500 nM T80975 CFYV96 44577766 IC50 = 560 nM T80975 CB6S8M 44577793 IC50 = 300 nM T80975 CT1Z7P 44577794 IC50 = 2100 nM T80975 CO3GT7 44577795 IC50 = 610 nM T80975 CF1Q2I 44577796 IC50 = 140 nM T80975 C1A5PZ 44577797 IC50 = 2000 nM T80975 CLER65 44577838 IC50 = 160 nM T80975 C4MKN8 44577839 IC50 = 540 nM T80975 CYPA37 44577840 IC50 = 730 nM T80975 CCZF36 44577841 IC50 = 2000 nM T80975 CR2C1B 44577875 IC50 > 10000 nM T80975 CD58EB 44577876 IC50 > 10000 nM T80975 CD78HT 44577877 IC50 = 1900 nM T80975 C8A2XU 44577878 IC50 = 660 nM T80975 CWS6V9 44577940 IC50 = 1000 nM T80975 CN7R2A 44577941 IC50 = 810 nM T80975 CZ0FO8 44577942 IC50 = 560 nM T80975 C43VMO 44577943 IC50 = 52 nM T80975 C1M8EI 44577985 IC50 = 355 nM T80975 C19SWX 44577986 IC50 > 10000 nM T80975 CY39BK 44577987 IC50 = 250 nM T80975 C92TQY 44577988 IC50 = 250 nM T80975 CAD1B9 44578019 IC50 = 830 nM T80975 CMJ5A4 44578020 IC50 > 10000 nM T80975 C3WYT4 44578021 IC50 > 10000 nM T80975 CL5O6H 44578022 IC50 = 7800 nM T80975 CXD9B4 44578561 IC50 = 6100 nM T80975 CTB96Y 44579918 IC50 = 18 nM T80975 C4Q1CA 44579956 IC50 = 5940 nM T80975 CF32AO 44579957 IC50 > 100000 nM T80975 C07YKU 44579993 IC50 > 100000 nM T80975 C3QLS4 44579994 IC50 > 100000 nM T80975 C7Q1VU 44580077 IC50 > 20000 nM T80975 CL90SE 44580358 IC50 > 20000 nM T80975 CK1VE7 44580420 IC50 = 6000 nM T80975 CH2R7X 44580449 IC50 > 20000 nM T80975 C1VH0C 44580532 IC50 > 20000 nM T80975 CXC52J 44580649 IC50 = 500 nM T80975 CE32BQ 44580689 IC50 = 800 nM T80975 C8Z5AX 44580778 IC50 > 20000 nM T80975 C14VTA 44581528 IC50 = 7600 nM T80975 CM75ND 44581529 IC50 > 25000 nM T80975 C6RJZ5 44581565 IC50 = 40 nM T80975 CE2C7W 44581602 IC50 = 250 nM T80975 C5WOE2 44586449 IC50 > 50000 nM T80975 C0VF8M 44586450 IC50 > 50000 nM T80975 C4K7NP 44586451 IC50 = 42300 nM T80975 C1JNR5 44586452 IC50 = 16800 nM T80975 C6T8UP 44586490 IC50 = 132100 nM T80975 CU95NI 44586526 IC50 > 200000 nM T80975 CBK9R3 44586527 IC50 > 200000 nM T80975 CA18IW 44586528 IC50 > 200000 nM T80975 C0YSZ2 44586577 IC50 = 24900 nM T80975 CGQR60 44586767 IC50 > 100000 nM T80975 CVRQ96 44586768 IC50 > 100000 nM T80975 C05HTO 44586769 IC50 = 4500 nM T80975 CX0R8V 44586770 IC50 = 13000 nM T80975 CQA2K1 44586794 IC50 = 77000 nM T80975 CH67VY 44586829 IC50 > 100000 nM T80975 C0HOF8 44586830 IC50 = 35000 nM T80975 C86ADQ 44586832 IC50 > 100000 nM T80975 CZAF65 44586833 IC50 > 100000 nM T80975 CWP37F 44586834 IC50 = 13000 nM T80975 CT5HM0 44586867 IC50 = 3200 nM T80975 CGK6C7 44586868 IC50 > 100000 nM T80975 C70DAO 44586869 IC50 = 9800 nM T80975 C2JIZ9 44586870 IC50 = 7800 nM T80975 CYU2G3 44586896 IC50 = 32000 nM T80975 C7G6KH 44586897 IC50 = 7000 nM T80975 C4L9BF 44586898 IC50 > 100000 nM T80975 CM45ZR 44586899 IC50 = 98000 nM T80975 CVU93G 44586900 IC50 > 100000 nM T80975 CMV3W2 44586901 IC50 > 100000 nM T80975 CV2W4P 44586928 IC50 > 100000 nM T80975 C95XRW 44586929 IC50 > 100000 nM T80975 CCT91D 44586930 IC50 = 2900 nM T80975 CJ4HT0 44587324 IC50 = 70000 nM T80975 CD56YX 44587325 IC50 = 31000 nM T80975 C4KW0O 44587326 IC50 = 17000 nM T80975 CX3O7R 44590991 IC50 = 1890 nM T80975 CBJ92M 44590992 IC50 = 790 nM T80975 CDG2S0 44590993 IC50 > 10000 nM T80975 CF78DX 44590994 IC50 > 10000 nM T80975 CKBN26 44590995 IC50 > 10000 nM T80975 CE91VG 44591030 IC50 = 150 nM T80975 CAI2X9 44591117 IC50 = 390 nM T80975 CD51XN 44591118 IC50 > 10000 nM T80975 CH0O2G 44591119 IC50 > 10000 nM T80975 C90IVK 44591355 IC50 = 4230 nM T80975 CE4G8R 44591356 IC50 > 10000 nM T80975 CN39VL 44591357 IC50 = 210 nM T80975 C5JYA9 44591358 IC50 > 10000 nM T80975 C7EOZ3 44591359 IC50 > 10000 nM T80975 C9WXA4 44591374 IC50 = 33 nM T80975 C9C8AH 44591375 IC50 = 770 nM T80975 C4E3NV 44591376 IC50 = 82 nM T80975 CUZG74 44591377 IC50 = 1150 nM T80975 C1JOA9 44591378 IC50 = 140 nM T80975 C9YV4O 44591404 IC50 = 210 nM T80975 C0AWD1 44591405 Ki = 70 nM T80975 C6EBW0 44591406 IC50 > 10000 nM T80975 C5XJ2N 44591407 IC50 = 770 nM T80975 CZ8F6B 44591439 IC50 = 230 nM T80975 CL7RC8 44591440 IC50 = 890 nM T80975 C0T1RY 44591441 IC50 = 1110 nM T80975 CL1TJ4 44591442 IC50 = 43 nM T80975 CQ9VS5 44591443 IC50 = 710 nM T80975 CY1A7W 44593407 IC50 = 294 nM T80975 C18QMJ 44595039 IC50 = 9.6 nM T80975 C28QLM 44605035 IC50 > 50000 nM T80975 C75XHS 44605037 IC50 > 50000 nM T80975 C8M5KI 44611919 IC50 = 19.1 nM T80975 CU3RF1 45139989 IC50 > 10000 nM T80975 CQGZ06 45139991 IC50 > 10000 nM T80975 CN65TK 45258773 IC50 = 287.28 nM T80975 C4S1PJ 45258774 IC50 = 184.53 nM T80975 CUS28K 45258871 IC50 = 169.17 nM T80975 C1TMO9 45258872 IC50 = 176.24 nM T80975 CS0JO2 45258873 IC50 = 453.41 nM T80975 C91BZJ 45258874 IC50 = 87.11 nM T80975 C8CRG0 45258875 IC50 = 107.23 nM T80975 CYL3D2 45258876 IC50 = 81.43 nM T80975 C13HGP 45258877 IC50 = 129.26 nM T80975 CN95PD 45258878 IC50 = 112.52 nM T80975 CH8NU3 45263527 IC50 = 6 nM T80975 C4UM6Y 45273507 IC50 > 10000 nM T80975 C2C8RH 45379202 IC50 > 100000 nM T80975 C5NB2X 45379203 IC50 > 100000 nM T80975 CT5BJ1 45379204 IC50 > 100000 nM T80975 CB41VP 45379205 IC50 > 100000 nM T80975 C2VUR3 45379340 IC50 > 100000 nM T80975 C8WXT4 45379341 IC50 > 100000 nM T80975 CQL29T 45379342 IC50 = 66000 nM T80975 CM7CB1 45379343 IC50 > 100000 nM T80975 C68WYX 45379344 IC50 = 140 nM T80975 C27MFU 45379345 IC50 = 400 nM T80975 C2O6VB 45379346 IC50 = 95 nM T80975 CLMB07 45379347 IC50 = 190 nM T80975 C8H5BL 45379490 IC50 = 330 nM T80975 C4YV6H 45379491 IC50 = 190 nM T80975 CRK4H3 45379492 IC50 = 80 nM T80975 CSM20A 45379493 IC50 = 290 nM T80975 CWP35H 45379494 IC50 = 130 nM T80975 CV2AZ7 45379495 IC50 = 51 nM T80975 CMP03L 45379496 IC50 = 6100 nM T80975 C6HM4U 45379605 IC50 = 57000 nM T80975 C6T1SW 45379606 IC50 = 530 nM T80975 CHNS21 45379607 IC50 = 35 nM T80975 C8HV1P 45379608 IC50 = 1200 nM T80975 CT6U7X 45379609 IC50 = 50 nM T80975 C5ATD8 45379610 IC50 = 28 nM T80975 C2APY4 45379611 IC50 = 52 nM T80975 CODU08 45379711 IC50 = 15 nM T80975 C79MTY 45379712 IC50 = 18 nM T80975 C8LMI5 45379713 IC50 = 11 nM T80975 CTJQ49 45379714 IC50 = 190 nM T80975 C15CVY 45379715 IC50 = 130 nM T80975 CM0P8B 45379716 IC50 = 99 nM T80975 C9XC4B 45379717 IC50 = 140 nM T80975 C1U6ST 45379811 IC50 = 87 nM T80975 CWB1C2 45379812 IC50 = 1500 nM T80975 CATM81 45379814 IC50 = 2000 nM T80975 C4W3OR 45379815 IC50 = 2600 nM T80975 C4KWJ3 45379956 IC50 = 48940 nM T80975 C2CU0B 45380067 IC50 = 27640 nM T80975 C6E2SC 45482700 IC50 > 10000 nM T80975 CZXH74 45482750 IC50 > 10000 nM T80975 C6C1JY 45488014 IC50 = 5 nM T80975 C4LI7T 45488043 IC50 = 200 nM T80975 C39YHU 45488044 IC50 = 30 nM T80975 C3XTH9 45488051 IC50 = 4 nM T80975 C4MH0A 45488054 IC50 = 10 nM T80975 C53DBE 45488073 IC50 = 89 nM T80975 CL5W8C 45488074 IC50 = 5 nM T80975 CN67YM 45488075 IC50 = 6 nM T80975 C8QIZ1 45488076 IC50 = 19 nM T80975 CZW27U 45488085 IC50 = 50 nM T80975 C96BNW 46179972 IC50 = 3.3 nM T80975 CNI92D 46182735 IC50 < 1 nM T80975 CH5VI6 46186825 IC50 = 10 nM T80975 C4A2MR 46190224 IC50 = 3900 nM T80975 CKX73S 46190225 IC50 = 330 nM T80975 CUA97D 46209401 IC50 = 160 nM T80975 CWN74L 46209503 IC50 = 5800 nM T80975 CKY01V 46209504 IC50 = 5100 nM T80975 CF57GK 46215462 IC50 = 8 nM T80975 CZ58FY 46215814 IC50 = 840 nM T80975 CZBL95 46220496 IC50 = 243 nM T80975 CMBJ68 46222580 IC50 = 660 nM T80975 C1GO2Y 46222581 IC50 = 150 nM T80975 CN8LX6 46224241 IC50 = 10 nM T80975 CPI8M7 46224242 IC50 = 66 nM T80975 C0TYK4 46224262 IC50 = 10 nM T80975 CXV0J1 46224334 IC50 = 6.2 nM T80975 CY3HW5 46224684 IC50 > 10000 nM T80975 C1U7IT 46225595 IC50 > 10000 nM T80975 C8YPN0 46225596 IC50 = 280 nM T80975 C34JTS 46225597 IC50 = 3300 nM T80975 CGD73B 46225598 IC50 > 10000 nM T80975 CRDY89 46225610 IC50 = 120 nM T80975 C0JMT8 46225611 IC50 = 690 nM T80975 CF0D5J 46225612 IC50 = 12 nM T80975 CLZ1O6 46225634 IC50 = 62 nM T80975 CT70DX 46225640 IC50 = 350 nM T80975 C6AJ5N 46225647 IC50 = 335 nM T80975 C38BFC 46225657 IC50 = 1200 nM T80975 C1B3KS 46225663 IC50 = 44 nM T80975 CU46XI 46225664 IC50 = 2500 nM T80975 CO3HS2 46225665 IC50 = 610 nM T80975 C2UV1S 46225666 IC50 > 10000 nM T80975 CX5B1G 46225667 IC50 = 2250 nM T80975 C2Q9OH 46225668 IC50 > 10000 nM T80975 C16LEO 46225679 IC50 = 6900 nM T80975 C8S4QA 46225688 IC50 = 250 nM T80975 C2P9QO 46228508 IC50 = 196 nM T80975 C6E5PY 46228822 IC50 = 1370 nM T80975 C3T8AM 46228951 IC50 = 200 nM T80975 CYZV41 46231219 IC50 = 82 nM T80975 C7J5UP 46231220 IC50 = 24.89 nM T80975 CC96GZ 46231221 IC50 = 22.5 nM T80975 CYT37A 46232443 IC50 = 23000 nM T80975 CG5K2H 46232509 IC50 > 50000 nM T80975 CA98UN 46232510 IC50 = 32000 nM T80975 CPK7Z8 46232511 IC50 = 26000 nM T80975 C8E4RB 46232512 IC50 > 50000 nM T80975 CZ52WR 46232513 IC50 > 50000 nM T80975 CAG90T 46232552 IC50 = 50000 nM T80975 C1O4DG 46232553 IC50 = 33000 nM T80975 CSHX24 46232554 IC50 > 50000 nM T80975 C48ZVW 46232555 IC50 = 11000 nM T80975 CTYB95 46232607 IC50 = 20 nM T80975 C5KMG3 46232608 IC50 = 20 nM T80975 CZ90EI 46232636 IC50 = 860 nM T80975 C7ON5A 46233287 IC50 > 10000 nM T80975 C9H4YO 46233889 IC50 = 130 nM T80975 CRT34L 46235770 IC50 = 11 nM T80975 CC2M1T 46831715 IC50 = 70700 nM T80975 C40JIK 46836783 IC50 = 3 nM T80975 C18YZM 46836784 IC50 < 10 nM T80975 CL2YG9 46836785 IC50 = 10 nM T80975 C0GA7Y 46836852 IC50 = 256 nM T80975 CL1E8Y 46836853 IC50 = 271 nM T80975 CF5J7R 46836854 IC50 < 10 nM T80975 CRQ61H 46836855 IC50 > 3000 nM T80975 C2DB9U 46836856 IC50 < 10 nM T80975 CX93NC 46836917 IC50 = 32 nM T80975 CFR1C6 46845026 IC50 = 100 nM T80975 CW0P5B 46845702 IC50 = 1500 nM T80975 C7KM0E 46845704 IC50 = 1010 nM T80975 CE3WH9 46865125 IC50 > 200000 nM T80975 C45LYT 46865445 IC50 > 200000 nM T80975 CO3P0J 46866604 IC50 < 50000 nM T80975 C1XEY4 46866615 IC50 > 200000 nM T80975 CF6K3E 46866616 IC50 > 200000 nM T80975 CX43UQ 46871756 IC50 = 2100 nM T80975 C5WC9K 46871765 IC50 = 2200 nM T80975 CQB16A 46872415 Ki > 4000 nM T80975 CLS29B 46872626 IC50 > 10000 nM T80975 CRS61F 46879438 IC50 = 135 nM T80975 C27JEF 46879439 IC50 = 1497 nM T80975 CF0T8P 46879440 IC50 = 1364 nM T80975 C12RMW 46879441 IC50 = 2094 nM T80975 CH2D7N 46879442 IC50 = 1113 nM T80975 CI6OD8 46879443 IC50 = 249 nM T80975 C7YD4Q 46879444 IC50 = 185 nM T80975 C8MN5Q 46879445 IC50 = 117 nM T80975 CX6SW2 46879446 IC50 = 245 nM T80975 CNF3V6 46879447 IC50 = 8181 nM T80975 CW46VY 46879448 IC50 = 133 nM T80975 CLK6X3 46879907 IC50 = 6365 nM T80975 C2A8KO 46880066 IC50 = 1748 nM T80975 CBRP80 46880067 IC50 = 1472 nM T80975 C3FY2B 46880068 IC50 = 599 nM T80975 CX89TY 46880069 IC50 = 1365 nM T80975 CB0XY1 46880070 IC50 = 318 nM T80975 CUD81V 46880071 IC50 = 941 nM T80975 CZP58Q 46880072 IC50 = 609 nM T80975 CC8OF9 46880073 IC50 = 549 nM T80975 CF41HG 46880098 IC50 = 296 nM T80975 C6O2YG 46880099 IC50 = 1015 nM T80975 CI78DM 46880100 IC50 = 17 nM T80975 CU04ZK 46880101 IC50 = 52 nM T80975 C4E0MF 46880133 IC50 = 92 nM T80975 COJ16A 46880134 IC50 = 464 nM T80975 C71MGJ 46880135 IC50 = 260 nM T80975 C3R6TL 46880213 IC50 = 516 nM T80975 CT8BQ4 46880214 IC50 = 8817 nM T80975 C0JTO4 46880215 IC50 = 10577 nM T80975 CAFN49 46880216 IC50 > 10000 nM T80975 C2O8RZ 46886323 IC50 = 29 nM T80975 CA57MX 46886970 IC50 = 45700 nM T80975 CRGH62 46886971 IC50 = 300 nM T80975 C68AGR 46886972 IC50 > 300000 nM T80975 CP32GW 46886973 IC50 = 85600 nM T80975 C48JWD 46886974 IC50 = 113100 nM T80975 C7H3MD 46887038 IC50 = 1400 nM T80975 C40NOR 46887039 IC50 > 300000 nM T80975 C7I4SB 46887074 IC50 = 27200 nM T80975 CI5QX2 46887110 IC50 > 300000 nM T80975 C0Q7NG 46887111 IC50 > 300000 nM T80975 CU15AN 46887112 IC50 > 300000 nM T80975 CD90BV 46887113 IC50 > 300000 nM T80975 CH3O9K 46887255 IC50 = 112300 nM T80975 C7NUT3 46887298 IC50 = 49400 nM T80975 CWV65D 46887299 IC50 = 22100 nM T80975 CH5BZ6 46887300 IC50 = 25200 nM T80975 C20UCB 46887348 IC50 = 57500 nM T80975 C0KEG5 46887349 IC50 = 40500 nM T80975 CY59RB 46887397 IC50 = 31600 nM T80975 CL5R0D 46888599 IC50 = 2830 nM T80975 C3IE0X 46888601 IC50 = 1060 nM T80975 C1A0XQ 46888603 IC50 = 2170 nM T80975 CB5YQ1 46888635 IC50 = 1220 nM T80975 C6YC4O 46888663 IC50 = 1170 nM T80975 C0AUT8 46888665 IC50 = 2030 nM T80975 CAZT96 46888666 IC50 > 50000 nM T80975 CS4U3P 46888668 IC50 = 1450 nM T80975 CASV10 46888710 IC50 = 940 nM T80975 CY2TV5 46888712 IC50 = 2180 nM T80975 CX5AL6 46888740 IC50 = 2070 nM T80975 CSWE93 46888742 IC50 = 27140 nM T80975 CCXK70 46888806 IC50 = 3000 nM T80975 C40DPT 46888807 IC50 = 1100 nM T80975 CZB8P0 46888808 IC50 = 1400 nM T80975 C7K9CZ 46888809 IC50 = 700 nM T80975 C0VSL7 46888810 IC50 = 1000 nM T80975 CIXV03 46888811 IC50 = 2500 nM T80975 C6UH7Y 46888812 IC50 = 5300 nM T80975 C84SJR 46888813 IC50 = 1400 nM T80975 CE1JL7 46889250 IC50 > 2000 nM T80975 COT4E8 46889251 IC50 > 20000 nM T80975 CQ27HK 46889273 IC50 = 1900 nM T80975 CHL36R 46889321 IC50 = 44 nM T80975 CA9J0L 46889322 IC50 = 149 nM T80975 COI7R4 46889323 IC50 < 50 nM T80975 CR8VH5 46889324 IC50 < 50 nM T80975 CJZC67 46889343 IC50 = 3 nM T80975 CZI7F3 46889344 IC50 = 16 nM T80975 CVK8I9 46889345 IC50 = 16 nM T80975 CVJ9X5 46889346 IC50 = 8 nM T80975 CTJ6L7 46889382 IC50 = 22 nM T80975 C4W7IC 46889383 IC50 = 9 nM T80975 C83AHJ 46889384 IC50 = 20 nM T80975 C9PZ4W 46889385 IC50 = 44 nM T80975 CGYT07 46889401 IC50 = 37 nM T80975 CMT73H 46889402 IC50 = 36 nM T80975 CAZ69B 46889403 IC50 = 65 nM T80975 CKP3D5 46889404 IC50 = 7 nM T80975 CB7SP1 46889850 IC50 = 5 nM T80975 CN19IK 46889851 IC50 < 10 nM T80975 CSQF75 46889884 IC50 = 6 nM T80975 CH8KA5 46889885 IC50 < 10 nM T80975 CP56KX 46889886 IC50 < 10 nM T80975 CW7AR1 46889887 IC50 = 10 nM T80975 CMNK35 46889911 IC50 = 10 nM T80975 CHW3Z2 46889912 IC50 = 77 nM T80975 CIV0K1 46889913 IC50 = 52 nM T80975 CST80X 46889914 IC50 < 50 nM T80975 CIZA86 46890251 IC50 = 1058 nM T80975 CM02UJ 46890253 IC50 = 1754 nM T80975 CB7VI8 46890254 IC50 = 10000 nM T80975 C7V3IA 46890314 IC50 = 2218 nM T80975 CHE6A1 46890315 IC50 = 48 nM T80975 C1YS5A 46890918 IC50 = 5400 nM T80975 CJ5S3N 46890968 IC50 = 690 nM T80975 CAGE32 46890969 IC50 = 2300 nM T80975 C3A7BP 46890970 IC50 = 5350 nM T80975 CTV73J 46890971 IC50 = 4100 nM T80975 CG35WP 46891025 IC50 = 130 nM T80975 C3FBH0 46891026 IC50 = 6000 nM T80975 CYOU90 46891080 IC50 = 1015 nM T80975 CJ16KH 46891081 IC50 = 8300 nM T80975 C7DOF4 46891082 IC50 = 1000 nM T80975 CRPL41 46891148 IC50 = 435 nM T80975 C6FJ7G 46891184 IC50 > 10000 nM T80975 C1B2UZ 46891185 IC50 = 9200 nM T80975 CYM5B2 46891226 IC50 = 500 nM T80975 C2DZE0 46891227 IC50 > 10000 nM T80975 C1W0JX 46891228 IC50 = 1900 nM T80975 CI3VZ0 46891275 IC50 = 7350 nM T80975 C0WYM1 46898022 IC50 = 10000 nM T80975 CTZ71Y 46898039 IC50 = 0.5 nM T80975 CB92VU 46912443 IC50 > 200000 nM T80975 CU6HC7 46912444 IC50 > 200000 nM T80975 C8A4KU 46912445 IC50 > 200000 nM T80975 CNOS56 46912446 IC50 > 200000 nM T80975 CV38NE 46912546 IC50 > 200000 nM T80975 CQLT07 46913878 IC50 < 1000 nM T80975 C60GAV 46929544 IC50 = 3270 nM T80975 CCN08S 46934144 IC50 = 33200 nM T80975 CJ4T3N 47120995 IC50 > 10000 nM T80975 C02SVR 49798997 IC50 = 10.2 nM T80975 C8DA5K 49798998 IC50 = 7.9 nM T80975 CO18QM 49798999 IC50 = 0.9 nM T80975 CC8FS1 49799031 IC50 = 30.6 nM T80975 CLNI64 49799032 IC50 = 4.7 nM T80975 CG7K2D 49799066 IC50 = 27 nM T80975 C27SKR 49799067 IC50 = 271.9 nM T80975 CCX04I 49799068 IC50 = 13.7 nM T80975 CQZC18 49799069 IC50 = 31.5 nM T80975 C2HA1O 49799301 IC50 = 10 nM T80975 C62OBF 49799302 IC50 > 1000 nM T80975 C1QC4V 49799333 IC50 > 1000 nM T80975 CG3LY7 49799334 IC50 > 1000 nM T80975 CZBW04 49799372 IC50 = 20.4 nM T80975 CN1M2D 49799373 IC50 = 22.1 nM T80975 CHIQ50 49799374 IC50 = 7.6 nM T80975 C45FZO 49799375 IC50 = 3.4 nM T80975 C0SJ7Q 49804868 IC50 > 5000 nM T80975 CHSF07 49806372 IC50 > 1000 nM T80975 COR4V2 49806718 IC50 = 3124 nM T80975 C5ME3S 49806721 IC50 > 5000 nM T80975 C67HGW 49806722 IC50 = 186 nM T80975 C8ML5D 49806794 IC50 > 12000 nM T80975 CY90BD 49818230 IC50 = 530 nM T80975 C2XZ8A 49830351 IC50 = 6 nM T80975 CGOR85 49830358 IC50 = 14 nM T80975 CJ3SU6 49830359 IC50 = 3 nM T80975 CKO52Y 49830360 IC50 = 15 nM T80975 CVS85M 49831162 IC50 = 240 nM T80975 C9L3XR 49838879 IC50 > 50000 nM T80975 C3ZI9B 49840051 IC50 > 10000 nM T80975 CDFE41 49840052 IC50 > 10000 nM T80975 C1XHO0 49840114 IC50 = 9500 nM T80975 CIMT03 49840186 IC50 > 10000 nM T80975 CIX4E3 49840245 IC50 > 10000 nM T80975 CLWN26 49840246 IC50 > 10000 nM T80975 CN89TG 49840317 IC50 = 600 nM T80975 C0AJ9R 49840318 IC50 = 600 nM T80975 CR58WT 49840391 IC50 = 2 nM T80975 CA2J6U 49840467 IC50 = 112 nM T80975 CB0S2P 49842666 IC50 = 1000 nM T80975 C0NA9U 49842670 IC50 > 100000 nM T80975 CC7MR2 49842671 IC50 = 93000 nM T80975 CAI20B 49842778 IC50 = 310 nM T80975 CRA74I 49842779 IC50 = 540 nM T80975 CF91RS 49843531 IC50 > 10000 nM T80975 C7A6IZ 49850211 IC50 = 600 nM T80975 C1BJ7D 49850390 IC50 = 827 nM T80975 C7JOA5 49850473 IC50 = 246 nM T80975 CB5O0I 49860186 IC50 = 7 nM T80975 C9W6SO 49860190 IC50 = 9 nM T80975 CQ3KU9 50899556 IC50 = 100 nM T80975 CK5TH3 50906783 IC50 = 910 nM T80975 C5RQ7C 50908680 Ki = 180 nM T80975 CD2K4R 50908681 Ki > 1000000 nM T80975 C2Y6QS 50938552 IC50 > 10000 nM T80975 C90ANW 50939489 IC50 = 370 nM T80975 C2Q0GE 50990922 IC50 = 40000 nM T80975 C61DVY 50990961 IC50 = 59 nM T80975 CV3UP9 50992247 IC50 = 6.2 nM T80975 CS9G6E 50997096 IC50 > 10000 nM T80975 CM42BY 51000510 Ki > 1000000 nM T80975 C9NYP4 51036677 IC50 > 10000 nM T80975 C4WRY3 51037112 IC50 > 10000 nM T80975 CRI28Z 51037948 IC50 > 10000 nM T80975 CDU4Q5 51346827 Ki > 8880 nM T80975 CTC8N1 51352971 IC50 = 28 nM T80975 C5QK8Y 51352972 IC50 = 78 nM T80975 CXA03W 52920796 IC50 = 340 nM T80975 CG5IK8 52936268 IC50 > 100000 nM T80975 CEQN27 52936621 Ki = 430 nM T80975 CM24LF 52938983 IC50 = 9.42 nM T80975 CYO5U4 52940598 IC50 = 1.202 nM T80975 CU72XM 52940665 IC50 = 112.6 nM T80975 CONY91 52940666 IC50 = 25.5 nM T80975 CU1P2L 52940797 IC50 = 12600 nM T80975 CI0DP3 52940860 IC50 = 0.1995 nM T80975 CS5OG1 52940980 IC50 = 19 nM T80975 CV52BN 52941091 IC50 > 10000 nM T80975 CL4I2K 52941234 IC50 = 9 nM T80975 C4R7IM 52941368 IC50 > 200000 nM T80975 C7S9UY 52941519 IC50 = 19 nM T80975 CH36PN 52941625 IC50 = 2.7 nM T80975 CBP18S 52941668 IC50 = 0.6026 nM T80975 C3LB5V 52941849 IC50 = 100 nM T80975 CNUE82 52941882 IC50 = 325.6 nM T80975 C39IPC 52942177 IC50 = 12 nM T80975 CDHJ08 52942235 IC50 = 100000 nM T80975 CG08LS 52942278 IC50 = 870 nM T80975 CG9E4A 52942446 Ki > 1000000 nM T80975 CM08KF 52942496 IC50 = 1400 nM T80975 CH7NE4 52942518 IC50 = 7.1 nM T80975 CN3H2J 52942791 IC50 = 8.9 nM T80975 CQA16I 52942852 IC50 = 4.4 nM T80975 C8SJ2Q 52942862 Ki > 1000000 nM T80975 C7BY6M 52942956 IC50 > 500000 nM T80975 CT8VW3 52943139 IC50 = 60 nM T80975 C1XEV2 52943394 IC50 = 1280 nM T80975 CSG8U1 52943668 IC50 = 4 nM T80975 C6R8AL 52943750 IC50 = 650 nM T80975 CH3FO1 52943828 IC50 = 4 nM T80975 CB56DX 52943829 IC50 = 7.6 nM T80975 CQ7ZL3 52944070 IC50 = 0.3715 nM T80975 CM0NA4 52944104 IC50 = 340 nM T80975 CA62KU 52944152 IC50 = 17800 nM T80975 CW2X5E 52944268 IC50 = 1 nM T80975 C1Q6RA 52944299 IC50 = 32.4 nM T80975 CFV1O5 52944388 IC50 = 0.5012 nM T80975 CKP62L 52944574 IC50 = 20 nM T80975 CIB62R 52944613 IC50 = 60 nM T80975 C40GQL 52944759 IC50 = 77 nM T80975 CLO46D 52944812 Ki = 2010 nM T80975 C4R3IB 52944922 IC50 = 230 nM T80975 CUDK18 52945153 IC50 = 61 nM T80975 CSK94T 52945251 IC50 = 32 nM T80975 CWPC54 52945348 IC50 = 2200 nM T80975 CQV34K 52945403 IC50 > 500000 nM T80975 C6L8WI 52945628 IC50 = 0.9 nM T80975 C4NLX7 52945630 IC50 = 100000 nM T80975 C9PX2J 52945752 IC50 = 10 nM T80975 CL4ED3 52945753 IC50 = 58 nM T80975 CZNE23 52945805 IC50 = 9.3 nM T80975 CXD6T8 52945845 IC50 = 100000 nM T80975 CV3SE7 52945860 IC50 = 1800 nM T80975 CU7A1G 52946083 IC50 = 6700 nM T80975 C0ADW5 52946084 IC50 = 4200 nM T80975 C6OI2Q 52946085 IC50 = 14 nM T80975 CU4Q1F 52946141 IC50 = 210 nM T80975 C95BXO 52946218 IC50 = 2.9 nM T80975 C9TD8F 52946373 IC50 = 6300 nM T80975 CA97SX 52946377 IC50 = 4.1 nM T80975 C17KVM 52946496 IC50 = 2.7 nM T80975 C97XZA 52946619 IC50 > 500000 nM T80975 CQWJ20 52946710 IC50 = 28.4 nM T80975 CX6Y5E 52946718 IC50 = 12.4 nM T80975 C9YQZ6 52946719 IC50 = 102.1 nM T80975 C7UZN1 52947137 IC50 = 940 nM T80975 C2WM9K 52947210 IC50 = 600 nM T80975 CYDN05 52947268 IC50 = 0.34 nM T80975 CJ5P3E 52947315 IC50 > 10000 nM T80975 CKH89Y 52947409 IC50 = 30 nM T80975 CE0X5U 52947574 IC50 > 200000 nM T80975 CSO9U5 52947605 IC50 = 3900 nM T80975 C57VIC 52947692 IC50 = 11 nM T80975 CD9S4I 52947801 IC50 > 500000 nM T80975 CA6IL3 52947802 IC50 > 500000 nM T80975 CAR09S 52947933 IC50 = 5.5 nM T80975 C1OLK2 52947942 IC50 = 23.4 nM T80975 CIR3Q0 52947964 IC50 > 10000 nM T80975 C9ZO1L 52948222 IC50 = 5.3 nM T80975 CZV6C3 52948268 IC50 = 21.88 nM T80975 C63VCY 52948336 IC50 = 23 nM T80975 CIPT89 52948377 IC50 = 9.7 nM T80975 CI6GX2 52948511 Ki = 300 nM T80975 C95EIM 52948533 IC50 = 3300 nM T80975 C1K9OJ 52948578 IC50 = 110 nM T80975 CNZ0E5 52948579 IC50 = 18 nM T80975 CPZA39 52948599 IC50 > 10000 nM T80975 C2KAJ4 52948634 IC50 = 89200 nM T80975 CT39LX 52948665 IC50 = 14 nM T80975 CE3WD7 52948666 IC50 = 3.8 nM T80975 C1VYU3 52948961 IC50 = 72.8 nM T80975 CSD23N 52949156 IC50 = 13.5 nM T80975 CL63KX 52949370 IC50 = 3.802 nM T80975 CFN2V3 52949618 IC50 = 9400 nM T80975 CWA74O 52949707 Ki = 470 nM T80975 C0A1GQ 52949915 IC50 = 116300 nM T80975 CIKY86 52949957 IC50 = 19 nM T80975 CL7K3V 52949960 IC50 = 9.4 nM T80975 C7G3YC 52950146 IC50 = 33 nM T80975 C2CT5J 53236670 IC50 > 100000 nM T80975 C3M6LV 53236671 IC50 > 100000 nM T80975 CZ5L6F 53239373 IC50 > 100000 nM T80975 C2WFI8 53239374 IC50 > 100000 nM T80975 C0ZHF8 53239375 IC50 > 100000 nM T80975 CD1EQ3 53239587 IC50 > 100000 nM T80975 CJ56EO 53244398 IC50 = 48 nM T80975 C64IQX 53244399 IC50 = 590 nM T80975 C1P3BC 53244475 IC50 = 373 nM T80975 C09SDH 53257410 IC50 > 10000 nM T80975 C2P3OT 53316977 IC50 = 4300 nM T80975 CVR3Y8 53317217 IC50 = 3410 nM T80975 C3RWG6 53317335 IC50 = 142 nM T80975 C4G6AW 53317731 IC50 > 10000 nM T80975 C9M5NX 53317732 IC50 = 2800 nM T80975 CE8OY2 53317913 IC50 < 1 nM T80975 CP97TR 53318517 IC50 = 2500 nM T80975 C42CVB 53318518 IC50 = 4500 nM T80975 CYM63Q 53318625 IC50 = 6.5 nM T80975 C8JS3Q 53318626 IC50 = 152 nM T80975 C1TFU9 53318931 Ki = 1.3 nM T80975 CK7W5F 53318958 IC50 = 1400 nM T80975 CZS8K4 53319042 Ki > 8880 nM T80975 C8E2OS 53319840 IC50 = 1100 nM T80975 C61COD 53319841 IC50 = 160 nM T80975 CL9K5W 53319941 IC50 > 100000 nM T80975 CP6HR7 53320237 Ki = 24 nM T80975 CUD21V 53320263 Ki > 8880 nM T80975 CZ0BV7 53320342 IC50 = 190 nM T80975 CX59LD 53320915 IC50 = 24000 nM T80975 CV19GL 53322464 IC50 = 3160 nM T80975 CNFW10 53322526 IC50 = 150 nM T80975 CZY0J7 53323592 IC50 = 2300 nM T80975 CESA85 53323614 Ki > 8880 nM T80975 C23RHN 53323819 IC50 > 10000 nM T80975 CMB7H4 53323821 IC50 > 10000 nM T80975 C3OYR7 53323909 IC50 = 180 nM T80975 C5KVH8 53324227 Ki = 328 nM T80975 CPLS09 53324303 IC50 > 10000 nM T80975 C2W9OA 53324451 IC50 = 5.8 nM T80975 CCKD48 53324892 IC50 = 82000 nM T80975 CFO5P2 53325089 IC50 = 2300 nM T80975 CO2L5V 53325090 IC50 = 300 nM T80975 CIPC27 53325139 IC50 = 5100 nM T80975 CE9D8O 53325140 IC50 = 4600 nM T80975 CBJM45 53326441 IC50 = 3100 nM T80975 CCBS06 53326481 IC50 = 2210 nM T80975 CT6E5C 53354781 IC50 = 182.3 nM T80975 CM7P3W 53357328 IC50 = 100 nM T80975 CE8OA7 53357593 IC50 = 290 nM T80975 C8NA4L 53384644 IC50 > 30000 nM T80975 CVG90B 53389651 IC50 > 10000 nM T80975 C8D9XG 53736592 IC50 > 10000 nM T80975 CKAP47 54578772 IC50 = 137 nM T80975 CR9F8Q 54578773 IC50 = 60.8 nM T80975 C4Z1NO 54578774 IC50 = 455 nM T80975 CD6RH1 54578996 IC50 > 5000 nM T80975 CV79SW 54578997 IC50 > 5000 nM T80975 CK1EM6 54580365 IC50 = 50 nM T80975 C4SN3X 54580366 IC50 = 30 nM T80975 C1HZ4Y 54581368 IC50 = 50 nM T80975 CA6H2U 54581369 IC50 = 5500 nM T80975 C5P9BQ 54581370 IC50 = 4300 nM T80975 CW7NH3 54582387 IC50 = 700 nM T80975 C7R4UG 54582388 IC50 = 600 nM T80975 C9SZ2I 54582389 IC50 > 10000 nM T80975 CO6B0E 54583043 IC50 > 10000 nM T80975 CL40KE 54583375 IC50 = 60 nM T80975 C2MFX7 54585296 IC50 = 6200 nM T80975 C3PGE2 54585958 IC50 > 10000 nM T80975 CV7HJ8 54585959 IC50 > 10000 nM T80975 CY4RH6 54586238 IC50 = 40 nM T80975 C8QA0M 54586239 IC50 > 10000 nM T80975 C47JTI 54586838 IC50 = 92 nM T80975 CL1I5C 54587267 IC50 = 5600 nM T80975 C1INS8 54597142 IC50 = 45 nM T80975 C0SC3J 54672928 IC50 = 25 nM T80975 CDMS75 54672929 IC50 = 21 nM T80975 CP5ZC3 54672931 IC50 = 72 nM T80975 C6OS4F 54672932 IC50 = 51 nM T80975 CR64QL 54673093 IC50 = 42 nM T80975 CE1D2H 54673094 IC50 = 64 nM T80975 CJL9T7 54673095 IC50 = 78 nM T80975 C73LSR 54673096 IC50 = 38 nM T80975 C3EJ0P 54673693 IC50 = 2385 nM T80975 CET93B 54673697 IC50 > 5000 nM T80975 C0JMY7 54673975 IC50 = 70100 nM T80975 C4XJR5 54675504 IC50 = 15 nM T80975 CE1ZK6 54759168 IC50 > 10000 nM T80975 C8AB1J 54759606 Ki = 3.8 nM T80975 C1XS2J 54760383 IC50 = 20 nM T80975 C9ZFS1 54764923 IC50 = 4950 nM T80975 CM8JX1 56604907 Ki = 7.8 nM T80975 CQ17GA 56640518 IC50 > 200000 nM T80975 CG20VK 56640520 IC50 > 200000 nM T80975 CZ9C8M 56640588 IC50 > 200000 nM T80975 CH0D7P 56640590 IC50 > 200000 nM T80975 CN9QD7 56643097 IC50 > 10000 nM T80975 CFJ37O 56649380 IC50 = 108 nM T80975 CV8B1X 56649401 IC50 = 72 nM T80975 CUEW30 56649402 IC50 = 28 nM T80975 CK2OT6 56649403 IC50 = 12 nM T80975 CVN1Z8 56649405 IC50 = 93 nM T80975 CPG0I4 56659823 IC50 > 1000 nM T80975 C4UPH5 56659824 IC50 = 200 nM T80975 CVDT38 56659825 IC50 > 1000000 nM T80975 C3A7HL 56663233 IC50 > 1000000 nM T80975 CY12ML 56663288 IC50 > 1000 nM T80975 CK53GA 56663289 IC50 = 410 nM T80975 CY2RD1 56663290 IC50 > 1000 nM T80975 C6XVT5 56666663 IC50 = 140 nM T80975 CKE5U3 56666717 IC50 = 560 nM T80975 C1HTO5 56670140 IC50 = 2720 nM T80975 CC3J1A 56673651 IC50 = 130 nM T80975 C4TD2Q 56673654 IC50 = 250 nM T80975 CGN54D 56676922 IC50 > 1000000 nM T80975 CU0M8W 56676973 IC50 = 70 nM T80975 CH5R3Q 56676974 IC50 > 1000 nM T80975 CUD53B 56676975 IC50 = 450 nM T80975 CO2GI9 56676977 IC50 > 1000000 nM T80975 CFS43O 56680303 IC50 > 1000 nM T80975 C5RK1U 56680304 IC50 > 1000 nM T80975 CVM7U4 56683624 IC50 = 160 nM T80975 CBW28D 56683625 IC50 > 1000 nM T80975 CT4E8R 56832546 IC50 = 6500 nM T80975 CR50TJ 56835147 IC50 = 5.5 nM T80975 CV5BM0 56835148 IC50 = 16 nM T80975 CRAJ75 56835149 IC50 = 17 nM T80975 CI5ZJ7 56835161 IC50 > 100000 nM T80975 C2ML5S 56837168 IC50 = 290 nM T80975 C87YOZ 56929808 IC50 = 320 nM T80975 CCW89V 56932477 IC50 = 237 nM T80975 CR3FK5 56932525 IC50 = 38 nM T80975 CS68GF 56933759 IC50 = 6580 nM T80975 CN7W4J 56935352 IC50 = 60 nM T80975 CY36EG 56945171 IC50 = 10 nM T80975 C4OG7H 56945172 IC50 = 56 nM T80975 CH0QA3 56945173 IC50 = 54 nM T80975 CM0NQ5 56945174 IC50 = 190 nM T80975 CXKF03 56945175 IC50 = 310 nM T80975 CE07AQ 56945176 IC50 = 1400 nM T80975 CU86KC 56945272 IC50 = 21 nM T80975 C9SX7F 56945273 IC50 = 1 nM T80975 CG7VH5 56945274 IC50 = 51 nM T80975 C6WU4V 56945277 IC50 = 10 nM T80975 CGLH06 56950183 IC50 = 63 nM T80975 CGQ94I 56950740 IC50 = 31000 nM T80975 CN1XL0 56950741 IC50 > 100000 nM T80975 C3ER0V 56950742 IC50 = 48000 nM T80975 CEZ14X 56950743 IC50 = 43000 nM T80975 CTL49B 56950878 IC50 = 87000 nM T80975 CM5HO1 56950881 IC50 = 2400 nM T80975 C9CLJ0 56950882 IC50 = 1200 nM T80975 CG0VC7 56950883 IC50 = 1900 nM T80975 CE1GO5 56950884 IC50 = 1400 nM T80975 CLQ4Z9 56950885 IC50 = 2600 nM T80975 C40BPN 56951005 IC50 = 1300 nM T80975 CL9XP2 56951006 IC50 = 2400 nM T80975 CKV5O2 56951007 IC50 = 210 nM T80975 C97QIR 56951008 IC50 = 27000 nM T80975 C7U9SL 56951304 IC50 = 5080 nM T80975 C0GQ9I 56951305 IC50 = 32100 nM T80975 C5YT6A 56951306 IC50 = 620 nM T80975 CB03EH 56951307 IC50 = 480 nM T80975 C2NJ4K 56951684 IC50 = 73.41 nM T80975 CRJ6H8 56953639 IC50 = 7200 nM T80975 C3D6YR 56953640 IC50 = 7250 nM T80975 CZ9F6B 56953642 IC50 = 5300 nM T80975 CTDR35 56953644 IC50 = 7400 nM T80975 CYF6D8 56953645 IC50 = 4800 nM T80975 CR20WU 56953646 IC50 = 4800 nM T80975 C86GAQ 56953648 IC50 = 9400 nM T80975 CMRB39 56953766 IC50 = 5700 nM T80975 CNG63B 56953767 IC50 = 5700 nM T80975 C1OC9P 56953892 IC50 = 7300 nM T80975 CF5AV8 56953893 IC50 = 4000 nM T80975 CBHG03 56953894 IC50 = 6800 nM T80975 CB5I7C 56953895 IC50 = 5000 nM T80975 C1NIS7 56954003 IC50 = 6800 nM T80975 CEKO58 56954004 IC50 = 5050 nM T80975 C7FP1R 56954005 IC50 = 5050 nM T80975 C0PY2A 56954006 IC50 = 500 nM T80975 CU1QF7 56954007 IC50 = 3300 nM T80975 CG9X1J 56954008 IC50 = 4900 nM T80975 CM9Z4I 56954009 IC50 = 850 nM T80975 CX1U4G 56954130 IC50 = 500 nM T80975 CG1VI6 56954131 IC50 = 850 nM T80975 CLR6J2 56954132 IC50 = 5200 nM T80975 C9OZ7N 56954133 IC50 = 5250 nM T80975 CLJC74 56954134 IC50 = 5550 nM T80975 CEWB79 56954135 IC50 = 7800 nM T80975 CY2GE9 56954136 IC50 = 6500 nM T80975 C5ATX6 56954232 IC50 = 4650 nM T80975 CU3T6F 56954234 IC50 = 6200 nM T80975 CMWK36 56954235 IC50 = 6900 nM T80975 CM9O5W 56954236 IC50 = 1000 nM T80975 C35JTA 56954323 IC50 = 6450 nM T80975 CI5MT0 56954324 IC50 = 5200 nM T80975 C06IDB 56954325 IC50 = 3350 nM T80975 CMT80I 56954326 IC50 = 6950 nM T80975 CE68LB 56954327 IC50 = 3700 nM T80975 CA43UF 56954328 IC50 = 6600 nM T80975 CC85JQ 56954429 IC50 = 7450 nM T80975 CP58NG 56954518 IC50 = 6 nM T80975 C7K1CZ 56954519 IC50 = 40 nM T80975 CH1X3R 56954520 IC50 = 4 nM T80975 CMS50D 56954621 IC50 = 6 nM T80975 C30ALB 56954622 IC50 = 2 nM T80975 CZN89G 56954623 IC50 = 8 nM T80975 CI7U1E 56954736 IC50 = 4300 nM T80975 C18BFU 56954737 IC50 = 6800 nM T80975 CO7D3X 56954739 IC50 = 5600 nM T80975 CRZ0M5 56954836 IC50 = 5000 nM T80975 C04JZF 56954837 IC50 = 6800 nM T80975 CH98NL 56954839 IC50 = 5050 nM T80975 CN06PL 56954840 IC50 = 500 nM T80975 CH0SG3 56954841 IC50 = 3300 nM T80975 C3MYG6 56954954 IC50 = 4900 nM T80975 C6WAD7 56954955 IC50 = 850 nM T80975 CZ82IH 56954956 IC50 = 650 nM T80975 CSBQ86 56954957 IC50 = 850 nM T80975 CIM60L 56954958 IC50 = 5200 nM T80975 C1LC4G 56955061 IC50 = 5550 nM T80975 C4OY1T 56955062 IC50 = 7800 nM T80975 CSJ6L7 56955063 IC50 = 6500 nM T80975 C1GA2O 56955275 IC50 = 3300 nM T80975 CT1KX9 56955277 IC50 = 3700 nM T80975 CAK91L 56955954 IC50 > 3600 nM T80975 CI6QE5 56970263 IC50 = 1.3 nM T80975 C62OJE 56970264 IC50 = 0.9 nM T80975 C7S9ER 56970466 IC50 = 2.3 nM T80975 CDS06V 56973548 IC50 = 630.96 nM T80975 CUAV97 56973549 IC50 = 1258.93 nM T80975 CI0K7Y 56973550 IC50 = 25.12 nM T80975 CPHX64 57325478 IC50 > 50000 nM T80975 CQ9BW4 57325479 IC50 > 50000 nM T80975 C1JLW8 57332840 IC50 = 1560 nM T80975 CD01JZ 57332841 IC50 = 6120 nM T80975 CCFK37 57332844 IC50 = 2050 nM T80975 CK1SR7 57332969 IC50 = 3310 nM T80975 C5TRE2 57332970 IC50 = 1600 nM T80975 C46TJK 57332974 IC50 = 11050 nM T80975 C09ZJY 57333095 IC50 = 8840 nM T80975 C91FTP 57339386 IC50 = 13 nM T80975 CI70CT 57345538 IC50 = 319 nM T80975 C4YFJ5 57384105 IC50 = 17900 nM T80975 CV9RW5 57384106 IC50 = 25700 nM T80975 CW9X3F 57386061 IC50 = 1.1 nM T80975 CSW5N7 57390857 IC50 = 23 nM T80975 C6J1MV 57390858 IC50 = 25 nM T80975 C76CTU 57390859 IC50 = 15 nM T80975 C8XGE1 57390860 IC50 = 17 nM T80975 C7Q2FR 57391239 IC50 = 129.56 nM T80975 CR4T2Y 57391283 IC50 = 22900 nM T80975 CBL74E 57392425 IC50 = 56700 nM T80975 CD29OE 57392674 IC50 = 87 nM T80975 CV54CQ 57392675 IC50 = 105 nM T80975 CAV4E0 57392912 IC50 = 112.26 nM T80975 CKVG97 57394105 IC50 < 1000 nM T80975 C0Z2NO 57394379 IC50 = 65 nM T80975 COE05G 57394380 IC50 = 98 nM T80975 CUK5X0 57394651 IC50 = 148.31 nM T80975 CZ6QS8 57394652 IC50 = 232.78 nM T80975 C3UHX0 57394704 IC50 > 5000 nM T80975 CG18LI 57394786 IC50 > 200000 nM T80975 CEDP89 57394787 IC50 = 14900 nM T80975 CP6W4C 57394879 IC50 = 23800 nM T80975 CVR13L 57394880 IC50 = 65300 nM T80975 C8W6IG 57395117 IC50 = 21900 nM T80975 C29ZPK 57395544 IC50 > 25000 nM T80975 CA4Q3Y 57395925 IC50 = 100 nM T80975 C63PVN 57396403 IC50 = 154.27 nM T80975 CB4FP0 57396404 IC50 = 561.29 nM T80975 CD7C4R 57396463 IC50 = 759 nM T80975 CLW12J 57396498 IC50 = 312.98 nM T80975 CUGP85 57396545 IC50 = 22900 nM T80975 CBUP96 57396646 IC50 = 113400 nM T80975 C4J6UZ 57397845 IC50 < 1000 nM T80975 CO9WX1 57398201 IC50 = 207.51 nM T80975 CJ2M8C 57398202 IC50 = 103.82 nM T80975 C8PH3X 57398203 IC50 = 261.88 nM T80975 CA57MF 57398204 IC50 > 1000 nM T80975 CPV50W 57398282 IC50 = 357.81 nM T80975 CM2UH9 57398315 IC50 > 50000 nM T80975 CXJ68F 57398331 IC50 = 64500 nM T80975 C14ANY 57398417 IC50 > 200000 nM T80975 C0BGR6 57399335 IC50 = 30 nM T80975 CG5J6M 57399603 IC50 = 237 nM T80975 CP0C9I 57399604 IC50 = 45 nM T80975 CV2U6Y 57399605 IC50 = 50 nM T80975 C2KQ6S 57399855 IC50 = 92.23 nM T80975 C79GAB 57399856 IC50 = 389.16 nM T80975 CX2UW6 57399904 IC50 > 5000 nM T80975 CE31FR 57399905 IC50 = 4210 nM T80975 CFIQ57 57399944 IC50 = 481.97 nM T80975 CLCE87 57401362 IC50 = 73 nM T80975 C4RDM3 57401625 IC50 = 139.36 nM T80975 CHV17A 57401626 IC50 = 129.54 nM T80975 CC4TI7 57401627 IC50 = 82.71 nM T80975 CMY0R5 57401628 IC50 = 267.27 nM T80975 C3E4MA 57401677 IC50 = 882 nM T80975 C0BA7P 57401686 IC50 = 485 nM T80975 CXSZ60 57403362 IC50 = 157.21 nM T80975 CP9Z4O 57403409 IC50 = 2521 nM T80975 CRU80Y 57403410 IC50 > 5000 nM T80975 CUXB78 57403456 IC50 = 189.07 nM T80975 C9EQX5 57403457 IC50 = 367.32 nM T80975 CTK29F 57403494 IC50 > 50000 nM T80975 CZSM95 57412684 IC50 > 10000 nM T80975 CN53XW 57428969 IC50 = 38.1 nM T80975 C9D5OH 57441057 IC50 = 80 nM T80975 CHV32A 57441068 IC50 = 640 nM T80975 CG3EN7 57505462 IC50 = 89 nM T80975 CW0RF4 57505467 IC50 = 1.2 nM T80975 C47WSH 57505488 IC50 = 1.8 nM T80975 CPEA97 57505491 IC50 = 4.7 nM T80975 C3HW1A 57505499 IC50 = 1.4 nM T80975 C6Q7PR 57505501 IC50 = 3.7 nM T80975 CE59QS 57505507 IC50 = 1.4 nM T80975 CV41XZ 57505509 IC50 = 12 nM T80975 CW3IV7 57505514 IC50 = 0.96 nM T80975 C1WLN0 57505517 IC50 = 25 nM T80975 CVG48T 57505518 IC50 = 1.3 nM T80975 CW9J1N 57505524 IC50 = 5200 nM T80975 CXT0W8 57505525 IC50 = 52 nM T80975 CQ6JE4 57505526 IC50 = 12 nM T80975 CPNA23 57505527 IC50 = 29 nM T80975 C8P6RD 57505528 IC50 = 7.1 nM T80975 C94GZX 57505530 IC50 = 1.3 nM T80975 CKD28T 57505535 IC50 = 5.1 nM T80975 CZY3O7 57505782 IC50 > 10000 nM T80975 C5XQ7G 57505784 IC50 = 18 nM T80975 C4T7PW 57523998 IC50 > 10000 nM T80975 C1Q7LS 57523999 IC50 = 213 nM T80975 CPS79I 57524088 IC50 = 8568 nM T80975 C0CJ8Z 57524184 IC50 = 2165 nM T80975 C8ICV2 57524400 IC50 = 75 nM T80975 CL72NQ 57524403 IC50 = 95 nM T80975 CAU0K1 57524478 IC50 = 91 nM T80975 C1XJ6U 57708543 IC50 = 1.1 nM T80975 C6T0XE 57708545 IC50 = 11 nM T80975 CRX82C 57708547 IC50 = 650 nM T80975 C9YXA3 57708552 IC50 = 12 nM T80975 CHL0X4 57708558 IC50 = 1.3 nM T80975 CRF8M0 57708566 IC50 = 1 nM T80975 CE3SA4 57708574 IC50 = 2.7 nM T80975 CHOB21 57749087 IC50 = 1.5 nM T80975 C73LPE 57749112 IC50 = 1.2 nM T80975 CH80LX 57749129 IC50 = 2 nM T80975 CM8AO9 57749178 IC50 = 3.1 nM T80975 CW1B7I 57749184 IC50 = 0.48 nM T80975 C73QPZ 57749213 IC50 = 1.9 nM T80975 CA14JW 57749237 IC50 = 3.7 nM T80975 CQ1NO9 57749289 IC50 = 1.6 nM T80975 CUL72T 57749346 IC50 = 2.1 nM T80975 C8R4FE 57991377 IC50 = 483.6 nM T80975 CD6ZP3 58009815 IC50 = 200 nM T80975 CWU1Y3 58009825 IC50 = 160 nM T80975 C8S6MY 58010054 IC50 = 90 nM T80975 CM1B4V 58010265 IC50 = 1000 nM T80975 CVK0G4 58056356 IC50 > 50000 nM T80975 C7HPC2 58268648 Ki = 207 nM T80975 CI37CQ 58394927 IC50 = 2600 nM T80975 C6KO0G 58395044 IC50 = 3700 nM T80975 C2I3QW 58486157 IC50 = 14000 nM T80975 C7ZKF5 58486186 IC50 = 9400 nM T80975 CBF7L4 58486208 IC50 > 5000 nM T80975 C51FBH 58486335 IC50 > 50000 nM T80975 C35FWX 58486367 IC50 > 10000 nM T80975 C8X6YE 58557497 IC50 = 720 nM T80975 C3F1TD 59175242 IC50 = 19 nM T80975 CT0VL3 59175570 IC50 = 160 nM T80975 C8HL0B 59175611 IC50 = 120 nM T80975 CPJ1X6 59176320 IC50 = 173 nM T80975 C3L4JY 59176329 IC50 = 53 nM T80975 CI8AL0 59176330 IC50 = 166 nM T80975 CDJQ62 59176336 IC50 = 77 nM T80975 C2WXU1 59176348 IC50 = 42 nM T80975 C5UQG8 59252136 IC50 = 214 nM T80975 CL6YV2 59262747 IC50 = 970 nM T80975 C4IBV1 59375998 IC50 = 1.1 nM T80975 CV8Q2D 59376002 IC50 = 9.4 nM T80975 CL3ND8 59376009 IC50 = 3.9 nM T80975 CC2AF9 59376012 IC50 = 4.3 nM T80975 CR7CG3 59376014 IC50 = 3 nM T80975 C60RIS 59376021 IC50 = 9.7 nM T80975 CT3Q5G 59376025 IC50 = 2.7 nM T80975 C97YSI 59376026 IC50 = 3.8 nM T80975 CEH5X6 59376027 IC50 = 1.1 nM T80975 C79EBT 59376032 IC50 = 8 nM T80975 C06DNI 59376037 IC50 = 2.6 nM T80975 C0XM7N 59376046 IC50 = 11.8 nM T80975 C70WCP 59376053 IC50 = 2.3 nM T80975 C5IHG9 59376058 IC50 = 1 nM T80975 CTK90V 59376059 IC50 = 112.4 nM T80975 C7ZY5I 59376061 IC50 = 24.6 nM T80975 CFT69X 59376062 IC50 = 167.2 nM T80975 C7D0BF 59376072 IC50 = 1.6 nM T80975 CD0RP7 59376074 IC50 = 15 nM T80975 C3HXC7 59376075 IC50 = 2.5 nM T80975 CAY6H8 59376079 IC50 = 25.7 nM T80975 CCX2W0 59376082 IC50 = 11.4 nM T80975 CSF3A7 59394005 IC50 = 30 nM T80975 C2XF4E 59394015 IC50 = 10.1 nM T80975 C17QBI 59394091 IC50 = 8 nM T80975 COFM73 59394146 IC50 = 5.8 nM T80975 CRY78K 59394153 IC50 = 280 nM T80975 CE7R6V 59394170 IC50 = 1 nM T80975 C0KBI8 59394176 IC50 = 5 nM T80975 CDU96X 59394177 IC50 = 245 nM T80975 C6B9LN 59394180 IC50 = 1 nM T80975 CQ43TB 59394183 IC50 = 4 nM T80975 CWE56B 59394184 IC50 = 8 nM T80975 CP34RY 59394193 IC50 = 26 nM T80975 CS94UC 59394203 IC50 = 7 nM T80975 CT6C3U 59394220 IC50 = 9.4 nM T80975 CJL85Z 59394228 IC50 = 7.9 nM T80975 CSE0L8 59394239 IC50 = 17.9 nM T80975 C9EYX0 59394267 IC50 = 89 nM T80975 C2L7IF 59394319 IC50 = 25.2 nM T80975 C8V2KU 59394332 IC50 = 114 nM T80975 C5IQ4P 59394335 IC50 = 9 nM T80975 CRLI45 59394364 IC50 < 3 nM T80975 CMR0B4 59394373 IC50 = 0.7 nM T80975 C3N4OB 59394395 IC50 = 2.5 nM T80975 CR51YF 59394398 IC50 = 4.1 nM T80975 CY9RB5 59394429 IC50 = 29 nM T80975 CF15EM 59394433 IC50 = 1720 nM T80975 CHXC24 59394467 IC50 = 30 nM T80975 C2WG6Z 59394482 IC50 = 66 nM T80975 CE02IH 59394496 IC50 = 230 nM T80975 CZK2L6 59394513 IC50 = 2.1 nM T80975 C8RE1T 59394521 IC50 = 2 nM T80975 CX8LE7 59394540 IC50 = 8.8 nM T80975 CJK08F 59394622 IC50 = 2 nM T80975 CND6M8 59394643 IC50 = 3 nM T80975 CC18YM 59394672 IC50 = 12.8 nM T80975 CO9G2C 59394679 IC50 = 273 nM T80975 CIFB80 59394686 IC50 = 12.8 nM T80975 C83FCQ 59394698 IC50 = 17.4 nM T80975 C7A5KZ 59394725 IC50 = 1 nM T80975 C0YP9D 59394733 IC50 = 18 nM T80975 CP9OT3 59394764 IC50 = 2.8 nM T80975 CXT56U 59454465 IC50 = 7.4 nM T80975 CZ24KM 59454479 IC50 = 33 nM T80975 C5GV2P 59454483 IC50 = 76 nM T80975 C7N3LA 59454484 IC50 = 70 nM T80975 CCH48T 59454492 IC50 = 15 nM T80975 C8DT3V 59454506 IC50 = 330 nM T80975 CP9A8T 59503659 IC50 = 253 nM T80975 C1MA6J 59503711 IC50 = 481 nM T80975 CX29EU 59503744 IC50 = 234 nM T80975 C2BGR6 59506918 IC50 = 340 nM T80975 C0KZ6L 59507002 IC50 = 300 nM T80975 C6EJ9G 59507062 IC50 = 410 nM T80975 CHQK85 59507068 IC50 = 510 nM T80975 C1E3OI 59598370 Ki = 309 nM T80975 CQ2UE7 59598391 Ki = 389 nM T80975 C5AEN1 59598393 Ki = 1630 nM T80975 CUA1F5 59598396 Ki = 257 nM T80975 C0O6ZX 59598404 Ki = 246 nM T80975 CBMH78 59598415 Ki = 325 nM T80975 CYNP39 59598421 Ki = 191 nM T80975 CU1ER8 59598432 Ki = 2830 nM T80975 C0L5DN 59598437 Ki = 708 nM T80975 CKVB01 59598456 Ki = 131 nM T80975 CXJ63M 59603829 IC50 = 15 nM T80975 CQEU96 59603842 IC50 = 3.5 nM T80975 CCX2Q5 59864465 Ki = 42 nM T80975 COH62U 60097413 IC50 > 10000 nM T80975 C1MR8Q 60097495 IC50 > 10000 nM T80975 COM48T 60154284 IC50 = 1000 nM T80975 CB7KE0 60154285 IC50 = 630.96 nM T80975 CO75BK 60154286 IC50 = 3981.07 nM T80975 CEF48W 60154326 IC50 = 6309.57 nM T80975 C2Y7JC 60154327 IC50 = 501.19 nM T80975 COU2B3 60154328 IC50 = 1000 nM T80975 CKM5E6 60154329 IC50 = 2511.89 nM T80975 CVE49A 60154330 IC50 = 125.89 nM T80975 C3BMS1 60154331 IC50 = 1584.89 nM T80975 CBU4I5 60154332 IC50 = 501.19 nM T80975 C03CFA 60154333 IC50 = 199.53 nM T80975 CLK0O6 60154334 IC50 = 1000 nM T80975 C34QJR 60154335 IC50 = 501.19 nM T80975 CXO1I8 60154336 IC50 = 501.19 nM T80975 CNZX63 60154337 IC50 = 15848.93 nM T80975 C3I4KJ 60154338 IC50 = 1258.93 nM T80975 CRB5D8 60154339 IC50 = 19952.62 nM T80975 CYI9F7 60154340 IC50 = 501.19 nM T80975 CLY46E 60154341 IC50 = 3162.28 nM T80975 CNS3Y1 60154342 IC50 = 125.89 nM T80975 C7CS4I 60154343 IC50 = 398.11 nM T80975 C46LSW 60154344 IC50 = 1584.89 nM T80975 CR60YI 60154345 IC50 = 1258.93 nM T80975 CSZA16 60155724 IC50 > 3600 nM T80975 C4SGZ6 60165992 IC50 = 85000 nM T80975 C98NOD 60165993 IC50 = 13400 nM T80975 C3WIX5 60165994 IC50 = 25000 nM T80975 C0G5WC 60165995 IC50 = 38000 nM T80975 CEQ07N 60166135 IC50 = 69000 nM T80975 CRV13A 60166136 IC50 > 100000 nM T80975 CLP62H 60166137 IC50 = 44000 nM T80975 C9X0ZC 60166139 IC50 = 3200 nM T80975 CWPZ07 60166141 IC50 = 7200 nM T80975 C7MLW5 60182318 IC50 = 0.2 nM T80975 CIP7B1 60182373 IC50 = 14 nM T80975 CQ6KV9 60182388 IC50 = 2040 nM T80975 C08VMZ 60198892 IC50 = 7 nM T80975 C4K8YJ 60198895 IC50 = 370 nM T80975 C5ZB2G 60199003 IC50 = 50 nM T80975 CN3W2C 60199004 IC50 > 1000 nM T80975 CTR58Y 60199005 IC50 = 7 nM T80975 CU79HD 60202383 IC50 = 848 nM T80975 C9ZCT2 62705065 IC50 > 1000 nM T80975 CW9CS2 62705327 IC50 = 40 nM T80975 CY5KC6 66550688 IC50 = 2990 nM T80975 C4K2VC 66550892 IC50 = 2620 nM T80975 C10AMI 66553589 IC50 > 10000 nM T80975 C9O4GF 66555232 IC50 = 1700 nM T80975 C7MD5X 66556536 IC50 = 1584.89 nM T80975 CL3EN2 66556938 IC50 = 290 nM T80975 C6A3TN 66759619 IC50 > 20000 nM T80975 CY36UH 66760355 IC50 > 20000 nM T80975 CE20FQ 66760840 IC50 = 650 nM T80975 CZ5JA1 66761050 IC50 = 19900 nM T80975 CP94KX 66761096 IC50 = 3400 nM T80975 CLQ51N 66761102 IC50 > 20000 nM T80975 C51XCV 66781377 IC50 = 28 nM T80975 C1GJX2 66781520 IC50 = 67 nM T80975 CN9SC4 66968949 IC50 = 0.14 nM T80975 C1HSE0 67035086 IC50 = 440 nM T80975 CWI6K5 67035106 IC50 > 10000 nM T80975 C38RGB 67035556 IC50 = 6600 nM T80975 CV3HW2 67035568 IC50 > 10000 nM T80975 CE49GC 67098566 Ki = 590 nM T80975 CT35MO 67127525 IC50 = 153 nM T80975 C0CL1R 67127737 IC50 = 169 nM T80975 C37NKO 67129970 IC50 > 10000 nM T80975 CK80LJ 67130050 IC50 = 8540 nM T80975 CQ97ZW 67161103 IC50 = 16 nM T80975 CNP52W 67163022 IC50 = 7 nM T80975 CA63QI 67219716 IC50 = 3100 nM T80975 CV63UL 67240318 IC50 > 10000 nM T80975 CLBP14 67405002 IC50 = 17 nM T80975 C6D3QJ 67448476 IC50 = 5600 nM T80975 CNT0W7 67468470 IC50 > 5000 nM T80975 CLD91A 67468733 IC50 > 5000 nM T80975 C3U7GQ 67469028 IC50 > 5000 nM T80975 CZC9M5 67469084 IC50 > 5000 nM T80975 CO6W9D 68004741 IC50 = 120 nM T80975 CB6U7F 68005465 IC50 = 210 nM T80975 CK83VI 68005486 IC50 = 3400 nM T80975 C1RJ7Y 68005600 IC50 = 1000 nM T80975 COX3U9 68005621 IC50 = 280 nM T80975 CEXN58 68005732 IC50 = 340 nM T80975 CSK4L6 68208633 IC50 = 560 nM T80975 C8I7GC 68293638 IC50 > 10000 nM T80975 CD56XK 68293660 IC50 > 10000 nM T80975 C3JE5H 68356029 IC50 = 17 nM T80975 CBIL54 68678227 IC50 > 10000 nM T80975 C7GRV2 68755406 IC50 > 10000 nM T80975 C8WZE0 68777669 IC50 = 693 nM T80975 COK9X0 68779704 IC50 = 264 nM T80975 C47JKD 68780376 IC50 = 1540 nM T80975 CC42HY 68780543 IC50 = 266 nM T80975 CZ2F5K 68780558 IC50 = 1 nM T80975 CWQP24 68780634 IC50 = 14 nM T80975 C71UOK 68780741 IC50 = 7 nM T80975 C6LY1M 68781121 IC50 = 12 nM T80975 C0G1NM 68781294 IC50 = 19 nM T80975 C62GYI 68781318 IC50 = 467 nM T80975 C60FTP 68781521 IC50 = 50 nM T80975 CJBW54 68781929 IC50 = 18 nM T80975 C8KP2A 68782417 IC50 = 19 nM T80975 CNEM15 68782426 IC50 = 6 nM T80975 CP5IF4 68782618 IC50 = 68 nM T80975 C5W7QY 68782756 IC50 = 89 nM T80975 C49PZJ 68782797 IC50 = 15 nM T80975 C8W5RV 68782804 IC50 = 2 nM T80975 CE84YM 68782852 IC50 = 922 nM T80975 CVML10 68783198 IC50 = 9 nM T80975 C76VIM 68783233 IC50 = 292 nM T80975 CE0YK8 68783378 IC50 = 329 nM T80975 CYE91N 68783396 IC50 = 2 nM T80975 C0Q4XO 68783521 IC50 = 3 nM T80975 C0HA8V 68783839 IC50 = 6 nM T80975 CDE57I 68854992 EC50 = 196 nM T80975 CRG14Q 68855406 EC50 = 24 nM T80975 CLY7I4 68971880 EC50 = 26 nM T80975 CM4WN5 68976126 EC50 = 4 nM T80975 C5DGR9 69036886 IC50 = 1445 nM T80975 C4BT3M 69037249 IC50 = 1.9 nM T80975 CCS20X 69063773 IC50 = 245 nM T80975 CWS02A 69268131 EC50 = 90 nM T80975 CPF8U9 69269522 EC50 = 104 nM T80975 CMPQ52 69271243 EC50 = 19 nM T80975 C2A7YP 69272308 EC50 = 24 nM T80975 CC5X9W 69272552 EC50 = 146 nM T80975 CB13CE 69272823 EC50 = 14 nM T80975 CM9RU2 69519173 IC50 = 1200 nM T80975 CECZ23 70654418 IC50 > 1000 nM T80975 CG50UJ 70654476 IC50 = 26 nM T80975 C4BS5T 70654492 IC50 = 120 nM T80975 CKP9E6 70654499 IC50 = 180 nM T80975 CAI3J4 70654537 IC50 = 12 nM T80975 CEXK08 70654539 IC50 > 1000 nM T80975 C5NDK0 70654558 IC50 = 54 nM T80975 C0AP6Q 70654571 IC50 > 1000 nM T80975 CRVS29 70654613 IC50 = 300 nM T80975 COV46X 70654614 IC50 = 370 nM T80975 CPF8W3 70654623 IC50 = 22 nM T80975 CVL6N9 70654642 IC50 = 28 nM T80975 CP0O5A 70654694 IC50 = 560 nM T80975 C9QS6O 70654709 IC50 = 92 nM T80975 C4INO3 70654745 IC50 = 50 nM T80975 CC0S3D 70654753 IC50 > 1000 nM T80975 C7F4DB 70654775 IC50 = 18 nM T80975 C4I8WO 70654805 IC50 = 73 nM T80975 C5LFG2 70654826 IC50 = 620 nM T80975 CA0UR2 70654830 IC50 = 12 nM T80975 CWE94C 70654840 IC50 = 480 nM T80975 C23AJO 70654866 IC50 = 100 nM T80975 CS6I4T 70654868 IC50 = 48 nM T80975 CGU2P6 70654923 IC50 > 1000 nM T80975 C59APG 70654958 IC50 = 310 nM T80975 C2LTI3 70654979 IC50 = 12 nM T80975 C6EK1V 70654997 IC50 = 240 nM T80975 CJAI19 70655010 IC50 = 220 nM T80975 CX3V5C 70655056 IC50 = 170 nM T80975 C49KEL 70655062 IC50 = 12 nM T80975 CW8XC7 70655063 IC50 > 1000 nM T80975 CUYK36 70655070 IC50 = 370 nM T80975 CNQ56Y 70657170 IC50 = 240 nM T80975 C2A4PE 70660513 IC50 = 31 nM T80975 CF92MK 70660523 IC50 > 1000 nM T80975 C7QL4R 70660524 IC50 = 100 nM T80975 C5U0EL 70661438 IC50 > 1000 nM T80975 C98FWB 70661441 IC50 = 38 nM T80975 C03CKB 70661448 IC50 = 100 nM T80975 CH6S7Q 70681377 IC50 = 3 nM T80975 CEB12M 70681395 IC50 = 2073 nM T80975 CH27DE 70681409 IC50 = 1277 nM T80975 CN29RI 70681410 IC50 > 9740 nM T80975 CUEO45 70681644 Ki = 78.9 nM T80975 CRE52C 70683471 IC50 = 25 nM T80975 CFN46P 70683472 IC50 = 1 nM T80975 CRA3I8 70683473 IC50 = 2 nM T80975 CXTS83 70683500 IC50 = 7 nM T80975 C81YOT 70683501 IC50 = 6 nM T80975 CG93IE 70683519 IC50 = 20 nM T80975 C59QUO 70683775 Ki = 702 nM T80975 C3RQ0D 70683776 Ki = 3350 nM T80975 CVFU50 70685579 IC50 = 6 nM T80975 C39GML 70685599 IC50 = 6 nM T80975 CXSN14 70685622 IC50 > 10000 nM T80975 CKCU42 70687611 IC50 = 5800 nM T80975 CL24MP 70687766 IC50 = 1919 nM T80975 C3O4UL 70688040 Ki > 6600 nM T80975 CYP97H 70688851 IC50 > 10000 nM T80975 CH30CI 70689776 IC50 = 25 nM T80975 C1CJ8S 70689777 IC50 = 4 nM T80975 C51DHN 70689791 IC50 > 690 nM T80975 C6ITV3 70689792 IC50 = 82 nM T80975 CCD49V 70689801 IC50 = 3 nM T80975 CMLY63 70689816 IC50 = 4 nM T80975 C08ASR 70689830 IC50 > 8690 nM T80975 CL0F7V 70690072 Ki = 343 nM T80975 C7I6QX 70690073 Ki = 519 nM T80975 C3MY9A 70690322 IC50 > 1000000 nM T80975 CFVS38 70690323 IC50 > 1000000 nM T80975 CTH7W5 70690324 IC50 = 10 nM T80975 CGA43T 70690710 IC50 = 190 nM T80975 CEQP73 70690935 IC50 > 10000 nM T80975 CI27NT 70690992 IC50 = 74 nM T80975 C4TF3G 70691955 IC50 > 10000 nM T80975 CTWD94 70691956 IC50 > 10000 nM T80975 CIK5N2 70691957 IC50 = 183 nM T80975 C8RZP3 70691958 IC50 = 23 nM T80975 C0XRC9 70691981 IC50 = 4819 nM T80975 C3OVZ0 70692216 Ki = 18.4 nM T80975 CLZ65T 70692217 Ki = 2240 nM T80975 CUT1L7 70693079 IC50 > 10000 nM T80975 C6U8HO 70693451 IC50 = 104 nM T80975 C4N6ZM 70693874 IC50 = 8900 nM T80975 C9RT8C 70693982 IC50 = 67 nM T80975 C2ZIB3 70693989 IC50 = 1 nM T80975 CA4DU8 70693990 IC50 = 3 nM T80975 C05FGA 70693991 IC50 = 3 nM T80975 C2X1KJ 70694006 IC50 = 20 nM T80975 C54VLD 70694007 IC50 = 3 nM T80975 CWM0K6 70695185 IC50 = 431 nM T80975 CA6HC7 70696091 IC50 = 2 nM T80975 C6O3SM 70696108 IC50 = 4773 nM T80975 CQIS80 70696112 IC50 = 6 nM T80975 CW5Z7B 70696113 IC50 = 2 nM T80975 C1U7FS 70696114 IC50 = 8 nM T80975 CUV36N 70696589 IC50 = 40 nM T80975 C23VCD 70988670 IC50 = 0.42 nM T80975 C1CQ6R 71450431 IC50 = 10 nM T80975 CNHZ80 71452610 IC50 = 22500 nM T80975 CEBO91 71452977 IC50 > 10000 nM T80975 CV78TK 71454499 IC50 = 90 nM T80975 CKT60L 71455860 Ki = 98 nM T80975 C7X4MD 71456750 IC50 > 25000 nM T80975 CIZA19 71459836 IC50 = 80000 nM T80975 CT3V7E 71461003 IC50 = 32 nM T80975 CVR7F1 71461211 IC50 = 14 nM T80975 C6E7JR 71492737 IC50 > 25000 nM T80975 CAW17X 71494057 IC50 > 25000 nM T80975 CDE4X6 71494225 IC50 > 25000 nM T80975 CQY31T 71498139 IC50 = 15.37 nM T80975 CB8ZX2 71510447 IC50 = 261.1 nM T80975 C1KC5A 71510707 IC50 = 63.2 nM T80975 CZ4M5S 71511128 IC50 = 102.6 nM T80975 C7Q4CA 71522447 IC50 = 8 nM T80975 CSM8Q3 71524871 IC50 = 4100 nM T80975 CQ34CK 71524919 IC50 = 3400 nM T80975 CZQ2S4 71524965 IC50 = 2100 nM T80975 C8A9IN 71525006 IC50 = 3200 nM T80975 C0M4LC 71525009 IC50 = 1830 nM T80975 C5OBF0 71525245 IC50 = 24100 nM T80975 CJX73B 71525246 IC50 > 200000 nM T80975 CCN90I 71525247 IC50 = 43600 nM T80975 CY6JA9 71525248 IC50 = 16700 nM T80975 CGQJ60 71525249 IC50 = 124500 nM T80975 CMKD15 71525283 IC50 > 200000 nM T80975 C3OJ6R 71525284 IC50 = 89300 nM T80975 CP5Q2U 71525285 IC50 = 125600 nM T80975 CZ8N0J 71525286 IC50 = 16700 nM T80975 CG31MI 71525287 IC50 = 150900 nM T80975 CCN01X 71547862 IC50 > 10000 nM T80975 C1NPL0 71552941 IC50 = 13310 nM T80975 CA4PS8 71552942 IC50 = 15960 nM T80975 C29ZRL 71575213 IC50 = 38 nM T80975 C12IXZ 71575543 IC50 = 11 nM T80975 CRX81Q 71575642 IC50 = 2250 nM T80975 C1BCX0 71579696 IC50 > 1000 nM T80975 CGK76E 71583411 IC50 = 123800 nM T80975 CB5WX0 71583412 IC50 = 30300 nM T80975 CI8K3T 71583527 IC50 = 13200 nM T80975 C6FGI0 71583528 IC50 = 38900 nM T80975 C3QGE7 71583529 IC50 = 86100 nM T80975 CS9HX7 71583530 IC50 = 192000 nM T80975 CQTZ32 71583531 IC50 = 47800 nM T80975 C0G5RS 71583532 IC50 = 21300 nM T80975 CVEY46 71583533 IC50 = 89100 nM T80975 CX6TR7 71583634 IC50 = 31200 nM T80975 CR15QP 71583635 IC50 = 41000 nM T80975 CZ31PU 71583657 IC50 > 10000 nM T80975 CN73PF 71615287 IC50 = 560 nM T80975 CXNG24 71622198 IC50 = 68 nM T80975 CY28UI 71627417 IC50 = 730 nM T80975 CB6LS5 71658742 IC50 = 300 nM T80975 CIN8Q2 71658743 IC50 > 1000 nM T80975 CEY10J 71658863 IC50 = 190 nM T80975 CC40FI 71658864 IC50 = 35 nM T80975 CN7TP5 71659100 IC50 = 82 nM T80975 C3AMG7 71659101 IC50 = 130 nM T80975 CD84KP 71659102 IC50 = 71 nM T80975 CS3Q2M 71659227 IC50 = 120 nM T80975 CYSZ68 71659355 IC50 = 38 nM T80975 CP9C1O 71678016 IC50 = 140 nM T80975 C1KL8U 71678017 IC50 = 120 nM T80975 CG39HK 71678357 IC50 = 560 nM T80975 C2XGC7 71678520 IC50 = 250 nM T80975 CO2G7N 71678692 IC50 = 170 nM T80975 CIH6U9 71678693 IC50 = 340 nM T80975 C3T1HM 71678864 IC50 > 10000 nM T80975 C1FAU8 71679855 IC50 = 690 nM T80975 CS62NH 71698376 IC50 = 191.9 nM T80975 CI8X1R 71698379 IC50 = 653 nM T80975 C3OS8U 71714087 IC50 = 8 nM T80975 C92AZQ 71714088 IC50 = 210 nM T80975 CN1Y9I 71714230 IC50 = 16 nM T80975 CM6NE9 71714231 IC50 = 6 nM T80975 CG28AP 71714232 IC50 = 5 nM T80975 C91CRY 71714233 IC50 = 87 nM T80975 C67HDT 71714234 IC50 = 83 nM T80975 CRS05F 71714235 IC50 = 3 nM T80975 CVC19T 71714373 IC50 = 7 nM T80975 CD5C8J 71714374 IC50 = 900 nM T80975 C51ISR 71714375 IC50 = 320 nM T80975 C5HJK2 71714376 IC50 = 20 nM T80975 C70SJV 71714377 IC50 = 60 nM T80975 C59UBD 71716995 IC50 > 10000 nM T80975 CXSI14 71718330 IC50 > 100000 nM T80975 C4NQ8L 71719650 IC50 = 5000 nM T80975 C1TM3P 71720141 IC50 > 100000 nM T80975 CD4WV8 71727539 IC50 = 1.2 nM T80975 CU83YL 71730951 IC50 = 750 nM T80975 C1TD4L 71731206 IC50 = 540 nM T80975 CLI52C 71732474 IC50 = 32 nM T80975 C7F3ZM 71736390 IC50 = 33 nM T80975 CKYO24 71736864 IC50 = 170 nM T80975 CU1IL6 71741204 IC50 > 100000 nM T80975 CN1GA3 71741327 IC50 > 100000 nM T80975 COS5D7 71741328 IC50 > 100000 nM T80975 C8PWZ0 71741329 IC50 > 100000 nM T80975 CT4XR9 71741332 IC50 > 100000 nM T80975 CMLF37 71814652 IC50 > 20000 nM T80975 CPNQ29 71814653 IC50 = 8200 nM T80975 CY21KG 71814654 IC50 = 760 nM T80975 CJ98FV 71814655 IC50 = 18300 nM T80975 C9GS6R 71814656 IC50 > 20000 nM T80975 C4Q6FE 71815105 IC50 = 1771.5 nM T80975 C1E4RK 71818600 IC50 = 120 nM T80975 CX78NJ 71818601 IC50 = 350 nM T80975 C8WZ1R 71818732 IC50 = 100 nM T80975 C4B7ZW 71818733 IC50 = 190 nM T80975 CCKL45 72191698 IC50 = 330.3 nM T80975 CB64IQ 72194525 IC50 = 35.1 nM T80975 CKR0I7 72558179 EC50 = 65 nM T80975 CQXZ13 72700883 Ki = 64 nM T80975 CYG95S 72707651 IC50 > 5000 nM T80975 CNP0V5 72707724 IC50 > 5000 nM T80975 CU4A5Q 72707728 IC50 > 5000 nM T80975 CZAM98 72707790 IC50 > 5000 nM T80975 CP13FK 72707853 IC50 > 5000 nM T80975 C9OQ2I 72710839 IC50 > 10000 nM T80975 CM1J8X 72723451 IC50 = 2.72 nM T80975 C60TUV 72737208 IC50 > 10000 nM T80975 CJ3WA6 72737404 IC50 > 10000 nM T80975 C1DMB4 72737557 IC50 = 7.1 nM T80975 CH8I6T 72737558 IC50 = 5.6 nM T80975 C52VCP 72737559 IC50 = 9 nM T80975 C6R8DI 72943374 IC50 = 527 nM T80975 C7IZU6 73054720 IC50 > 300 nM T80975 CJ19NP 73054721 IC50 > 300 nM T80975 C06GET 73054722 IC50 = 17.5 nM T80975 CXQ0T5 73054723 IC50 = 12.8 nM T80975 CHZ0F2 73055002 IC50 = 179 nM T80975 C16PXZ 73055003 IC50 > 300 nM T80975 C3DC9R 73055004 IC50 = 4.06 nM T80975 CLDG01 73055005 IC50 > 300 nM T80975 C6MUI2 73055006 IC50 = 128 nM T80975 C3LZ8Q 73055289 IC50 = 4.55 nM T80975 C2CVD6 73055290 IC50 = 5.26 nM T80975 C9LC3E 73055291 IC50 = 12.8 nM T80975 COTU30 73055293 IC50 = 23.8 nM T80975 C4P1ZR 73055591 IC50 = 71.4 nM T80975 CE9S7A 73055592 IC50 = 16.7 nM T80975 CIX21U 73055593 IC50 = 17.6 nM T80975 CN5I9P 73055594 IC50 > 300 nM T80975 CV2T0U 73055595 IC50 = 69.9 nM T80975 CR6X3J 73055890 IC50 = 23.9 nM T80975 C3LSR9 73055891 IC50 = 33.3 nM T80975 C01PAZ 73055893 IC50 > 300 nM T80975 CF5LG4 73055894 IC50 = 14.3 nM T80975 CL3DZ7 73056170 IC50 = 40.9 nM T80975 CI37NA 73056171 IC50 = 129 nM T80975 C5PO4E 73056172 IC50 = 3.07 nM T80975 CS24KQ 73345824 IC50 = 15848.93 nM T80975 C8SIL6 73349435 IC50 = 531.9 nM T80975 CV21FR 73349643 IC50 = 50 nM T80975 CQ04OK 73350400 IC50 = 4100 nM T80975 C9TMA1 73352657 IC50 = 30 nM T80975 C7F0YR 73353451 IC50 = 85 nM T80975 CAV7T4 73354894 IC50 = 26200 nM T80975 CJ82UZ 73354897 IC50 = 45200 nM T80975 CZN1Y6 73354960 IC50 = 27 nM T80975 C6UA4K 73356522 IC50 > 3000 nM T80975 CYQ8K1 73357210 IC50 = 8 nM T80975 C2PAK9 73438493 IC50 = 21 nM T80975 C3UC9H 73891099 IC50 = 320 nM T80975 CBAT06 76071144 IC50 = 24 nM T80975 CW5OG2 76310006 IC50 > 100000 nM T80975 CV8QX0 76310169 IC50 = 26400 nM T80975 C32DZE 76310260 IC50 = 202 nM T80975 C2O6TS 76311163 IC50 = 2890 nM T80975 CI8H9X 76311164 IC50 = 3870 nM T80975 CVU96Q 76311165 IC50 = 2160 nM T80975 C7MLX4 76313718 IC50 = 23400 nM T80975 CRV24X 76313719 IC50 > 100000 nM T80975 C9RDO6 76314767 IC50 = 4890 nM T80975 COP50L 76314768 IC50 = 7210 nM T80975 C3I7UA 76314769 IC50 = 3400 nM T80975 CZK2V6 76317238 IC50 > 100000 nM T80975 CKG8C3 76317239 IC50 = 26900 nM T80975 CRO31B 76318365 IC50 = 2230 nM T80975 CA95JI 76318366 IC50 = 5370 nM T80975 CGYM87 76318367 IC50 = 2660 nM T80975 C73RZA 76318368 IC50 = 1090 nM T80975 C8P6KY 76322048 IC50 = 52500 nM T80975 C8JRL6 76322049 IC50 = 3170 nM T80975 CPD3W5 76324607 IC50 = 850 nM T80975 CA5L4W 76324771 IC50 > 30000 nM T80975 C4BSA5 76324834 IC50 = 15 nM T80975 C25ORT 76325670 IC50 = 3290 nM T80975 CPZN18 76328168 IC50 > 100000 nM T80975 C9GO0P 76328313 IC50 = 5960 nM T80975 C7OHZ4 76328389 IC50 = 51.2 nM T80975 CPXE65 76328390 IC50 = 170 nM T80975 C1G4OV 76328399 IC50 = 215 nM T80975 C38HPS 76329233 IC50 = 8570 nM T80975 CB5RH9 76329234 IC50 = 3480 nM T80975 C9J6FO 76329235 IC50 = 2030 nM T80975 CN18KC 76329236 IC50 = 1090 nM T80975 C9PDY0 76332896 IC50 = 3270 nM T80975 C2JUZ1 76332897 IC50 = 6740 nM T80975 CAP7F0 76335418 IC50 = 43300 nM T80975 C51LIY 76335419 IC50 > 100000 nM T80975 C39FTZ 76335685 IC50 = 3660 nM T80975 CT84NC 76336503 IC50 = 4960 nM T80975 CTO57P 76336504 IC50 = 1030 nM T80975 C4SQ2V 76336505 IC50 = 6450 nM T80975 CH8W7D 77461036 IC50 > 1000 nM T80975 CH4OV1 77631108 EC50 = 160 nM T80975 CWG4T2 78209992 IC50 = 156 nM T80975 CA65HB 78319164 IC50 = 200 nM T80975 C5U8VI 78426332 IC50 = 11.7 nM T80975 CE9R4L 78426885 IC50 = 40.1 nM T80975 CN0X2A 78427023 IC50 = 215.8 nM T80975 C4VUP1 78427168 IC50 = 68.5 nM T80975 CHLR89 78673838 IC50 = 6 nM T80975 CX93GA 85470895 IC50 = 10 nM T80975 C2WLZ6 85827467 Ki = 2760 nM T80975 CV8UZ1 86278565 IC50 = 2270 nM T80975 CSH3G2 86287525 IC50 = 72 nM T80975 C0GQ8S 86291490 IC50 = 79.1 nM T80975 CRQO23 86293280 IC50 = 997 nM T80975 C4OC7T 86293469 IC50 = 1035 nM T80975 CCJ43A 86302281 IC50 > 10000 nM T80975 CB5NJ4 86302541 IC50 = 1.5 nM T80975 CPJ25O 86302563 IC50 = 21.3 nM T80975 CPG3A5 86302574 IC50 > 30000 nM T80975 C08WGI 86566799 IC50 = 65.42 nM T80975 CWZ41G 86566934 IC50 = 110.2 nM T80975 C0ALG3 86567077 IC50 = 108.1 nM T80975 CW40TZ 86567079 IC50 = 21.8 nM T80975 CEY30N 86567080 IC50 = 89.9 nM T80975 C3I5JQ 86567457 IC50 = 63.5 nM T80975 C1BZA4 86567460 IC50 > 100 nM T80975 C5S7BY 86567464 IC50 = 2.5 nM T80975 C1Z8UJ 86567604 IC50 = 5.5 nM T80975 CZ0L3H 86567605 IC50 = 91.4 nM T80975 C1C5PN 86567669 IC50 = 2.6 nM T80975 CLO6A7 86567670 IC50 = 6.5 nM T80975 CUNA57 88876306 IC50 = 31 nM T80975 CDW95X 88876318 IC50 = 15 nM T80975 CE6RY9 88876331 IC50 = 53 nM T80975 CT1L6U 88876351 IC50 = 43 nM T80975 C31EBZ 88876355 IC50 = 25 nM T80975 CVEA94 88876366 IC50 = 15 nM T80975 CLE48M 89434293 IC50 = 279.9 nM T80975 C1HW4B 89735655 IC50 = 11000 nM T80975 C7TJR3 89814000 IC50 = 1900 nM T80975 C4WP7D 89827799 IC50 = 750 nM T80975 CV64KY 90183363 IC50 > 10000 nM T80975 CL4JO2 90183809 IC50 = 1990 nM T80975 CR1N0E 90367910 IC50 = 16 nM T80975 C81AZQ 90644555 IC50 = 50.1 nM T80975 C1J2ZY 90644557 IC50 = 40.6 nM T80975 CWNK43 90644559 IC50 = 30.1 nM T80975 CX39PY 90644653 IC50 = 1.9 nM T80975 C3PVN7 90644654 IC50 = 1.4 nM T80975 C8ODA6 90644655 IC50 = 18.2 nM T80975 CU5GC2 90644656 IC50 = 3.8 nM T80975 CBC7R8 90644657 IC50 = 10.8 nM T80975 C8HU6C 90644658 IC50 = 2.1 nM T80975 CFPN87 90644659 IC50 = 7.1 nM T80975 C4K5PJ 90644660 IC50 = 2.5 nM T80975 CIY9L5 90644661 IC50 = 2.6 nM T80975 CORH73 90644662 IC50 = 2.8 nM T80975 CM4X6B 90644663 IC50 = 3.1 nM T80975 CLO01U 90644664 IC50 = 3.3 nM T80975 C12GOF 90644665 IC50 = 6.1 nM T80975 C60KYR 90644666 IC50 = 24 nM T80975 CKZ4J7 90644667 IC50 = 4.5 nM T80975 CFQG67 90644668 IC50 = 5.7 nM T80975 CKF0T5 90644669 IC50 = 6.1 nM T80975 C5GO6S 90644670 IC50 = 7 nM T80975 C6A0LQ 90644671 IC50 = 7 nM T80975 CLYH98 90644672 IC50 = 7.1 nM T80975 CDU48F 90644673 IC50 = 7.3 nM T80975 CO3I8G 90644674 IC50 = 9.2 nM T80975 CO41EM 90644675 IC50 = 20.2 nM T80975 CS39GA 90644676 IC50 = 26.7 nM T80975 C5ORK2 90644677 IC50 = 40.8 nM T80975 COR98Y 90644938 IC50 = 16 nM T80975 C07COR 90644939 IC50 = 14 nM T80975 CDZ5R6 90644940 IC50 = 30.3 nM T80975 CAP53K 90644941 IC50 = 61.5 nM T80975 CT9C6L 90644942 IC50 = 54 nM T80975 CWT52M 90644943 IC50 = 219.9 nM T80975 CUCN60 90644944 IC50 = 4 nM T80975 C7Z2LF 90644945 IC50 = 46.6 nM T80975 CM8JV5 90644946 IC50 = 6.1 nM T80975 C7K3FV 90644947 IC50 = 5.6 nM T80975 CNVW64 90644948 IC50 = 12.7 nM T80975 CY13SF 90644949 IC50 = 43 nM T80975 CAZO78 90644950 IC50 = 9.8 nM T80975 CQ71IN 90644951 IC50 = 48 nM T80975 CE3SB9 90644952 IC50 = 83.6 nM T80975 CNH6P4 90644953 IC50 = 44.5 nM T80975 CQ5I8Z 90644955 IC50 = 52 nM T80975 C4DY8K 90644956 IC50 = 24.5 nM T80975 CD52AH 90644957 IC50 = 255.6 nM T80975 CHV49F 90644958 IC50 = 181 nM T80975 C6T9IR 90644959 IC50 = 230 nM T80975 C8GH1V 90644960 IC50 = 4394 nM T80975 CXO2R8 90644961 IC50 = 196.2 nM T80975 C0K7FY 90644962 IC50 = 2716 nM T80975 C4IO7C 90644963 IC50 = 2468.5 nM T80975 CJ21KA 90644964 IC50 = 55 nM T80975 C8F3XR 90644965 IC50 = 16 nM T80975 C5S3YB 90645165 IC50 = 425.42 nM T80975 CY0UC4 90645194 IC50 > 10000 nM T80975 C6Q4DH 90645475 IC50 = 8.5 nM T80975 C89HTB 90645476 IC50 = 34.4 nM T80975 CL32MR 90645477 IC50 = 50.3 nM T80975 C9ASG1 90645478 IC50 = 10.6 nM T80975 COY53U 90645479 IC50 = 76.3 nM T80975 C48OSQ 90645480 IC50 = 15.6 nM T80975 CL8GW5 90645481 IC50 = 66.2 nM T80975 CL7SC6 90645482 IC50 = 102.1 nM T80975 C5U6RM 90645483 IC50 = 58.2 nM T80975 CI3OD6 90645484 IC50 = 43.1 nM T80975 CCS47U 90645485 IC50 = 32.2 nM T80975 CXEB69 90645486 IC50 = 70.2 nM T80975 CX29IY 90655145 IC50 > 10000 nM T80975 CS3PJ0 90655410 IC50 = 52000 nM T80975 CMH6T8 90664306 IC50 = 1000 nM T80975 CP34KC 90664681 IC50 = 1260 nM T80975 CK3IS4 90664930 IC50 = 2120 nM T80975 CRL86F 90665697 IC50 > 1000 nM T80975 C9V6FU 90666397 IC50 > 1000 nM T80975 C5Q8VO 90666398 IC50 > 1000 nM T80975 CIB1E8 90666399 IC50 > 1000 nM T80975 C08ANK 90666400 IC50 > 1000 nM T80975 CL0KH2 90666401 IC50 > 1000 nM T80975 C9XI3E 90666402 IC50 > 1000 nM T80975 CLF29C 90666403 IC50 = 390 nM T80975 CU9XB7 90666404 IC50 = 190 nM T80975 CCL19D 90666405 IC50 = 180 nM T80975 CYVM38 90666406 IC50 = 36 nM T80975 CMY4T0 90666407 IC50 = 37 nM T80975 CNE54X 90666408 IC50 = 860 nM T80975 CA5KJ0 90667006 IC50 = 5.77 nM T80975 C54VAR 90667007 IC50 = 1.28 nM T80975 C10IDP 90667008 IC50 = 203 nM T80975 C6H3CS 90667009 IC50 = 7.01 nM T80975 C9KPW7 90667010 IC50 = 4.08 nM T80975 CJ0TR8 90667012 IC50 = 1.08 nM T80975 CJ2P9T 90667014 IC50 = 3.9 nM T80975 CR3M4F 90667015 IC50 = 9.87 nM T80975 CHDO09 90667016 IC50 = 3.77 nM T80975 CN8ZC3 90667017 IC50 = 8.9 nM T80975 CBAM42 90667697 IC50 = 9900 nM T80975 C3TCZ8 90667699 IC50 = 5400 nM T80975 C1M7UL 90667701 IC50 = 9200 nM T80975 C7J0CF 90667703 IC50 > 10000 nM T80975 CU5I7B 90667705 IC50 > 10000 nM T80975 CH16WR 90667707 IC50 = 900 nM T80975 C8SX2E 90667875 IC50 = 400 nM T80975 CS73QB 90667877 IC50 = 500 nM T80975 CSM40E 90667879 IC50 = 800 nM T80975 CAZD95 90667881 IC50 = 300 nM T80975 CGU4Q0 90667883 IC50 = 500 nM T80975 CN1L2V 90667885 IC50 > 10000 nM T80975 C96DTL 90682879 IC50 = 20.2 nM T80975 C18ZOV 90718764 IC50 = 23 nM T80975 CT2GU1 91246771 IC50 = 24 nM T80975 CRF65D 91899696 IC50 = 10300 nM T80975 C0Y8ZK 91933875 IC50 > 1000 nM T80975 CAU45T 91971978 IC50 > 30000 nM T80975 C8F7XO 92131166 IC50 = 96.68 nM T80975 C4CE3S 94146587 IC50 = 20410 nM T80975 CPGV73 101884319 IC50 > 2000 nM T80975 CA1TZ3 101884321 IC50 > 2000 nM T80975 CG9KE7 101884322 IC50 > 2000 nM T80975 C84MVD 101884325 IC50 = 1400 nM T80975 CRI0S4 101891768 IC50 = 1660 nM T80975 C6D9CA 101896448 IC50 > 1000 nM T80975 C2VFS6 101898750 IC50 = 20 nM T80975 CK72FW 102129497 IC50 = 70.41 nM T80975 C5HRO7 102431711 IC50 = 23000 nM T80975 CV9S8Q 118111994 IC50 > 10000 nM T80975 C5QW0Y 118111995 IC50 > 10000 nM T80975 CH6M2V 118112005 IC50 = 280 nM T80975 CRL0O1 118112011 IC50 > 10000 nM T80975 CGI47W 118112014 IC50 = 1000 nM T80975 CU25TZ 118112016 IC50 = 4100 nM T80975 C4QB8Y 118112024 IC50 > 10000 nM T80975 C0KO2J 118112026 IC50 > 10000 nM T80975 CHCI59 118112037 IC50 > 10000 nM T80975 CAD76E 118112040 IC50 = 230 nM T80975 CWU3S7 118112047 IC50 = 2500 nM T80975 C29BPV 118112051 IC50 > 10000 nM T80975 CS06EV 118112055 IC50 > 10000 nM T80975 C4VBY7 118112056 IC50 > 10000 nM T80975 CYEO57 118112076 IC50 = 770 nM T80975 C8AE2F 118112077 IC50 > 10000 nM T80975 CD61JA 118112079 IC50 > 10000 nM T80975 CBA4O8 118112080 IC50 > 10000 nM T80975 CM1E5A 118112082 IC50 > 10000 nM T80975 CJ94NF 118112083 IC50 > 10000 nM T80975 C2AQ6Y 118112087 IC50 > 10000 nM T80975 C5QAZ7 118112091 IC50 > 10000 nM T80975 CNO0T7 118112099 IC50 > 10000 nM T80975 CH84RT 118112100 IC50 > 10000 nM T80975 CU6MI0 118112101 IC50 > 10000 nM T80975 C02OVL 118112108 IC50 = 5700 nM T80975 C7ACP6 118112114 IC50 = 1100 nM T80975 C5FT9N 118112115 IC50 > 10000 nM T80975 C4B1FL 118112118 IC50 > 10000 nM T80975 CT6A1B 118112122 IC50 > 10000 nM T80975 CTK8O1 118112125 IC50 > 10000 nM T80975 C0S9QW 118112133 IC50 = 5600 nM T80975 C0SQ7Y 118112144 IC50 > 10000 nM T80975 CR58UD 118112154 IC50 = 5900 nM T80975 CO3WA5 118112158 IC50 > 10000 nM T80975 C23GBT 118112186 IC50 = 230 nM T80975 C5HB0N 118112191 IC50 > 10000 nM T80975 CE9ZN0 118112194 IC50 > 10000 nM T80975 COD73Q 118112202 IC50 > 10000 nM T80975 C0TMZ8 118167692 IC50 > 5000 nM T80975 CU02NF 118559124 IC50 = 3 nM T80975 CY7BI2 118706214 IC50 > 10000 nM T80975 C1RO4V 118709802 IC50 = 830 nM T80975 CUD8S3 118709803 IC50 = 9350 nM T80975 CZ0NL4 118709804 IC50 = 6570 nM T80975 C2ZYH1 118709805 IC50 = 4760 nM T80975 C46SBZ 118709806 IC50 > 10000 nM T80975 CPE61B 118709808 IC50 = 8690 nM T80975 C3U5XI 118709809 IC50 = 6350 nM T80975 CV8Z3F 118709810 IC50 = 820 nM T80975 CGT82L 118709811 IC50 = 8700 nM T80975 C4INY8 118709812 IC50 = 1580 nM T80975 CHR4E5 118709813 IC50 = 90 nM T80975 C6P4YN 118709814 IC50 = 380 nM T80975 C0FU6Y 118709815 IC50 > 10000 nM T80975 CRT83K 118709816 IC50 > 10000 nM T80975 CX1TZ3 118709817 IC50 = 8850 nM T80975 C4H8VY 118709818 IC50 > 10000 nM T80975 CRVP89 118709819 IC50 = 760 nM T80975 C12WRM 118709820 IC50 = 1840 nM T80975 CAS3B5 118709821 IC50 = 8520 nM T80975 CF2YR1 118710237 IC50 = 20.7 nM T80975 C5X1PO 118710876 IC50 = 2480 nM T80975 C1RDB6 118710877 IC50 > 10000 nM T80975 CS9BU1 118710878 IC50 = 6800 nM T80975 C97POE 118710879 IC50 = 4650 nM T80975 CNC15F 118710880 IC50 > 10000 nM T80975 C2FYQ1 118710882 IC50 = 5490 nM T80975 CELA12 118710883 IC50 > 10000 nM T80975 C1WC7A 118710884 IC50 = 3520 nM T80975 CM3Q9F 118710885 IC50 = 1360 nM T80975 C0Z9YX 118710886 IC50 > 10000 nM T80975 CG1R6U 118710887 IC50 = 2400 nM T80975 CKA28F 118710888 IC50 = 240 nM T80975 C6JY4C 118710889 IC50 = 180 nM T80975 COU9E3 118710890 IC50 > 10000 nM T80975 C7B3WV 118710893 IC50 > 10000 nM T80975 C54MDP 118710894 IC50 > 10000 nM T80975 C3YA0S 118710895 IC50 = 8350 nM T80975 CKH4D1 118710896 IC50 = 30 nM T80975 CA2EK1 118710897 IC50 = 80 nM T80975 CPA4M3 118710898 IC50 = 7820 nM T80975 C4AHL2 118711367 IC50 > 10000 nM T80975 CWO9B7 118715995 IC50 = 560 nM T80975 C46QUT 118717614 IC50 > 200000 nM T80975 CJC34Y 118717615 IC50 > 200000 nM T80975 CFEP93 118717616 IC50 > 200000 nM T80975 CEC4H0 118717617 IC50 > 200000 nM T80975 CU2TG3 118717618 IC50 > 200000 nM T80975 C5OL0W 118717619 IC50 > 200000 nM T80975 CI5W9H 118720010 IC50 = 3290 nM T80975 COQ9S4 118720011 IC50 = 2240 nM T80975 C3KLI5 118723185 IC50 = 2300 nM T80975 CRQY80 118723194 IC50 = 1000 nM T80975 C7JYP8 118723210 IC50 = 56000 nM T80975 CI6QA2 118723212 IC50 = 2200 nM T80975 CZVH46 118725690 IC50 = 18600 nM T80975 C6GQL2 118725758 IC50 = 23400 nM T80975 C9KYM5 118727105 IC50 = 69.4 nM T80975 CN09QM 118727106 IC50 = 182.82 nM T80975 C2Q9ED 118727107 IC50 = 4.38 nM T80975 CL29HV 118727108 IC50 = 15.04 nM T80975 CA62YT 118727110 IC50 = 9.41 nM T80975 CU5I1L 118727112 IC50 = 130.17 nM T80975 C59QKO 118727113 IC50 = 22.85 nM T80975 CMI3B8 118727114 IC50 = 94.69 nM T80975 CUGV93 118727115 IC50 = 624.66 nM T80975 CCHR07 118727117 IC50 = 359.63 nM T80975 CQ0U5D 118727118 IC50 = 31.98 nM T80975 C8OQN9 118727119 IC50 = 214.87 nM T80975 CT7O5B 118727120 IC50 = 62.52 nM T80975 CDRW84 118727121 IC50 = 54.26 nM T80975 C4AW3V 118727122 IC50 = 14.48 nM T80975 CN04JV 118727123 IC50 = 2.02 nM T80975 CCW5L9 118727124 IC50 = 8.74 nM T80975 C5YX3Z 118727125 IC50 = 4.86 nM T80975 CDJ6R9 118727126 IC50 = 44.32 nM T80975 C7Q8NV 118727127 IC50 = 129.25 nM T80975 C9B8VT 118727129 IC50 = 85.32 nM T80975 C7D5ZY 118727130 IC50 = 27.58 nM T80975 C1ISD2 118727131 IC50 = 158.46 nM T80975 CMVE97 118727132 IC50 = 17.85 nM T80975 C65BYE 118727134 IC50 = 77.45 nM T80975 CAE08L 118727135 IC50 = 125.82 nM T80975 CQD5J1 118727136 IC50 = 71.89 nM T80975 CX9NY6 118727137 IC50 = 344.61 nM T80975 CHT6K9 118728811 Ki > 4000 nM T80975 CUA3Y2 118728812 Ki > 4000 nM T80975 CDQ78G 118728813 Ki > 4000 nM T80975 CZ6XL7 118728814 Ki > 4000 nM T80975 CMO67K 118728815 Ki > 4000 nM T80975 CR2M0Q 118728816 Ki > 4000 nM T80975 C62SCL 118728817 Ki > 4000 nM T80975 CSB30C 118728819 Ki = 1900 nM T80975 CV7XU8 118728820 Ki = 2400 nM T80975 C3J1EX 118728821 Ki > 4000 nM T80975 CIWB78 118728822 Ki > 4000 nM T80975 CP18SE 118728823 Ki = 2000 nM T80975 CM42CA 118728824 Ki > 4000 nM T80975 C9Q7CL 118728825 Ki > 4000 nM T80975 CCR3S0 118728826 Ki = 1500 nM T80975 CWYF91 118729842 IC50 = 32.3 nM T80975 CR54XL 118729843 IC50 = 18.6 nM T80975 CF3X9J 118729844 IC50 > 300 nM T80975 CT3Q6C 118729845 IC50 = 19.9 nM T80975 C1QWK6 118729846 IC50 = 6.7 nM T80975 CWUA61 118729847 IC50 = 5.8 nM T80975 C63CDP 118729848 IC50 = 20.9 nM T80975 C1WB7L 118729849 IC50 > 300 nM T80975 C8A7ZT 118729850 IC50 = 33.2 nM T80975 C9WDF4 118729851 IC50 = 38.5 nM T80975 CT08EZ 118729852 IC50 = 121.3 nM T80975 C25ODS 118731589 IC50 = 23 nM T80975 CT98EI 118731590 IC50 = 120 nM T80975 C9IZR4 118731591 IC50 = 36 nM T80975 C8U0ZH 118737468 IC50 = 2.38 nM T80975 CX1IU7 118753064 IC50 > 30000 nM T80975 CI93JD 118893305 IC50 = 365.9 nM T80975 C0UT7G 122177477 IC50 = 0.46 nM T80975 CSF49R 122177478 IC50 = 25 nM T80975 C08KEM 122179540 IC50 = 4100 nM T80975 C3AJ4C 122179546 IC50 = 6500 nM T80975 CG0RP7 122179547 IC50 = 1000 nM T80975 C1A0SQ 122179548 IC50 = 5000 nM T80975 CDTA86 122180042 IC50 = 0.36 nM T80975 CJ0D2O 122180043 IC50 > 200 nM T80975 CF5P9Y 122180044 IC50 = 4.6 nM T80975 C71CZL 122180045 IC50 = 63.08 nM T80975 CF58IL 122180047 IC50 > 200 nM T80975 CIR0T9 122180049 IC50 = 2.19 nM T80975 C0VG4X 122180050 IC50 = 0.22 nM T80975 CV1H5X 122180051 IC50 = 722.38 nM T80975 C9PWN1 122180053 IC50 > 1000 nM T80975 CF95BV 122180054 IC50 > 1000 nM T80975 C54XEN 122180056 IC50 > 1000 nM T80975 CSX35A 122180058 IC50 = 13.26 nM T80975 CZP2R3 122180059 IC50 > 1000 nM T80975 C9MNQ0 122180062 IC50 > 1000 nM T80975 C0GKH6 122180063 IC50 = 99.58 nM T80975 CWL85C 122180064 IC50 = 0.15 nM T80975 CJK5N8 122180065 IC50 = 0.14 nM T80975 C42GSX 122180520 Ki > 4000 nM T80975 CS85CU 122181413 IC50 = 29 nM T80975 CJ4T5W 122181414 IC50 = 170 nM T80975 CK8L4D 122181415 IC50 = 210 nM T80975 CQS67B 122181416 IC50 = 9000 nM T80975 CB2AG9 122181417 IC50 = 1200 nM T80975 CFET49 122181418 IC50 = 6600 nM T80975 CQU14E 122181419 IC50 = 90 nM T80975 CN81HR 122181799 IC50 = 160 nM T80975 C2D8UA 122181800 IC50 = 10 nM T80975 CMU6G9 122181801 IC50 = 55 nM T80975 C8DJ3K 122181802 IC50 = 170 nM T80975 CR9FQ7 122181803 IC50 = 120 nM T80975 CTS2C6 122181804 IC50 > 1000 nM T80975 CWA94G 122182409 IC50 = 92.6 nM T80975 CB0QF4 122183083 IC50 = 4800 nM T80975 CB2VY7 122183099 IC50 = 1000 nM T80975 CZ1U4R 122183100 IC50 = 960 nM T80975 C6VE0K 122185734 IC50 = 34 nM T80975 C9AVI2 122185735 IC50 = 59 nM T80975 C5JVK8 122185736 IC50 = 122 nM T80975 C9OWX5 122186256 IC50 = 343 nM T80975 C3J6BA 122186261 IC50 = 284 nM T80975 CEB0W5 122188019 IC50 > 100000 nM T80975 CJO0S7 122188020 IC50 > 100000 nM T80975 CAH78S 122188021 IC50 > 100000 nM T80975 CEX84Y 122188022 IC50 = 94 nM T80975 C6JBE0 122188023 IC50 = 107 nM T80975 C23VQA 122188024 IC50 = 206 nM T80975 C92INA 122188025 IC50 = 28 nM T80975 CEA7K6 122188026 IC50 = 11 nM T80975 CGB36N 122188027 IC50 = 15 nM T80975 CA17VG 122188028 IC50 = 16 nM T80975 C2EC9M 122188029 IC50 = 1160 nM T80975 C58SKJ 122188123 IC50 = 1390 nM T80975 C45LBH 122188124 IC50 = 8360 nM T80975 CE82JM 122188125 IC50 = 988 nM T80975 C6AQ8E 122188126 IC50 = 1947 nM T80975 CZN2V0 122188510 IC50 = 191 nM T80975 C4X7SD 122192466 IC50 = 2458 nM T80975 C5W8KA 122193537 IC50 = 2700 nM T80975 CB6M4T 122193759 IC50 = 3820 nM T80975 C65XUZ 122193760 IC50 > 10000 nM T80975 CHF47Y 122193761 IC50 = 3140 nM T80975 C1XHI4 122193762 IC50 = 12 nM T80975 CNX0Q2 122193763 IC50 = 91 nM T80975 CWV0C3 122193764 IC50 = 1160 nM T80975 CSG98Y 122193765 IC50 = 310 nM T80975 C1SED2 122193766 IC50 = 600 nM T80975 CINA05 122193767 IC50 = 710 nM T80975 C27WGV 122193768 IC50 = 1140 nM T80975 CCLQ75 122193769 IC50 = 8 nM T80975 CXDR48 122193770 IC50 = 18 nM T80975 C96LDU 122193771 IC50 = 16 nM T80975 C50HEA 122193772 IC50 = 9 nM T80975 CPA8C5 122193773 IC50 = 11 nM T80975 CM3G0Y 122193774 IC50 > 50000 nM T80975 CVM68S 122193775 IC50 > 50000 nM T80975 C0OLT4 122193776 IC50 = 17500 nM T80975 CU8Q7L 122193777 IC50 > 50000 nM T80975 C83XVM 122193778 IC50 > 50000 nM T80975 CIS0B2 122193779 IC50 > 50000 nM T80975 C26POY 122193780 IC50 = 5600 nM T80975 C59RDU 122193840 IC50 = 34 nM T80975 CXE87R 122193841 IC50 = 15 nM T80975 C17POX 122195140 IC50 = 28 nM T80975 CVA5O9 122195141 IC50 > 500000 nM T80975 CBC8W5 122195142 IC50 = 62 nM T80975 CIOC59 122195143 IC50 = 53000 nM T80975 CJ2EM4 122195144 IC50 = 5400 nM T80975 C3Z2PI 122195145 IC50 = 51900 nM T80975 C7I9NV 122195146 IC50 = 160 nM T80975 C7L0DH 122195147 IC50 = 37700 nM T80975 C9GHO4 122195148 IC50 > 500000 nM T80975 C19VJU 122195149 IC50 = 8400 nM T80975 CY75HQ 122195150 IC50 > 500000 nM T80975 CI6K8U 122195151 IC50 > 500000 nM T80975 C38ZUF 122195152 IC50 > 500000 nM T80975 C3Q1PE 122195153 IC50 > 500000 nM T80975 CSW97B 122195154 IC50 > 500000 nM T80975 C2T7WS 122195155 IC50 > 500000 nM T80975 CT3UK8 122195156 IC50 > 500000 nM T80975 CR06ZU 122195157 IC50 = 4700 nM T80975 C7NTI2 122195158 IC50 = 14900 nM T80975 CEG45A 122195159 IC50 = 53.6 nM T80975 CLF93A 122195160 IC50 = 59.2 nM T80975 CCI6S3 122195161 IC50 = 2.15 nM T80975 CGN15D 122195162 IC50 = 116 nM T80975 C0WUF7 122195163 IC50 = 0.5 nM T80975 CWV0R1 122195164 IC50 = 2.36 nM T80975 CO6AS1 122195165 IC50 = 2.28 nM T80975 C1R7NK 122195166 IC50 = 331 nM T80975 CAYW84 122195167 IC50 = 21 nM T80975 CD8ZR1 122195168 IC50 > 500 nM T80975 CA1S8F 122195169 IC50 > 500 nM T80975 C1Q3TI 122195170 IC50 = 205 nM T80975 CKF92Z 122195171 IC50 = 117 nM T80975 CJ4X6Q 122195172 IC50 = 41.8 nM T80975 CG1DW6 122195173 IC50 = 0.79 nM T80975 CK2I4M 122195174 IC50 > 500 nM T80975 CW9V2E 122195472 IC50 = 1.38 nM T80975 CNL26X 122195473 IC50 > 500 nM T80975 CBFG20 122195474 IC50 = 3.47 nM T80975 CG9R5W 122195476 IC50 > 100000 nM T80975 C2BM0D 122195480 IC50 > 100000 nM T80975 CN61IM 122195481 IC50 = 42000 nM T80975 CS71XH 122195525 IC50 = 476 nM T80975 C3AY9G 122195526 IC50 = 352 nM T80975 C2ZY0G 122195527 IC50 = 613 nM T80975 CFYL41 122195528 IC50 = 501 nM T80975 CS0NH6 122195529 IC50 = 625 nM T80975 C9JPK0 122195530 IC50 = 434 nM T80975 CEJB32 122195531 IC50 = 415 nM T80975 CFZ54V 122195532 IC50 = 462 nM T80975 CNOC04 122195533 IC50 = 370 nM T80975 CV2ZX8 122195534 IC50 = 138 nM T80975 C1LZB0 122195535 IC50 = 115 nM T80975 CW1HK5 122195536 IC50 = 84 nM T80975 C2K4OG 122195537 IC50 = 1260 nM T80975 CH79VD 122195538 IC50 = 2140 nM T80975 CZ9P8V 122195539 IC50 = 5200 nM T80975 CR6Q2V 122195540 IC50 = 2450 nM T80975 CG1H5X 122377977 IC50 = 1.6 nM T80975 CLM7K3 122604539 IC50 > 10000 nM T80975 C01JHI 122604566 IC50 > 10000 nM T80975 C8YA0F 122628813 IC50 = 240 nM T80975 COC02I 122629035 IC50 = 160 nM T80975 CY30FL 123752658 IC50 = 48.7 nM T80975 CZAY93 124197376 IC50 = 565 nM T80975 CZFG57 124197588 IC50 > 1000 nM T80975 C2LAM7 126591927 IC50 = 96 nM T80975 CE89QB 127024882 IC50 = 2480 nM T80975 C1WH5M 127024973 IC50 = 455 nM T80975 CUF81C 127025156 IC50 = 364.14 nM T80975 CP3LK5 127025157 IC50 = 21.57 nM T80975 C8QKX6 127025158 IC50 = 128.15 nM T80975 C86RIQ 127025203 IC50 = 1990 nM T80975 CR3KZ0 127025430 IC50 = 400 nM T80975 CWG54Q 127025431 IC50 = 2380 nM T80975 CDQ52G 127025443 IC50 > 500 nM T80975 CN3J0U 127025710 IC50 = 3110 nM T80975 C1DCG7 127025711 IC50 = 1440 nM T80975 C8KXV1 127025843 IC50 > 1000 nM T80975 C43JUF 127026070 IC50 = 376 nM T80975 C4HW8S 127027008 IC50 > 10000 nM T80975 C1EW7J 127027019 IC50 = 857 nM T80975 CT3Y6R 127027064 IC50 = 220 nM T80975 CI42FJ 127027065 IC50 = 313 nM T80975 CB2F4S 127027091 IC50 = 524 nM T80975 CO3A7W 127027092 IC50 = 270 nM T80975 C90VAW 127027093 IC50 = 832 nM T80975 CO9I6S 127027094 IC50 = 685 nM T80975 CFY28V 127027095 IC50 = 364 nM T80975 CGE73Y 127027096 IC50 = 182 nM T80975 CBT52X 127027296 IC50 = 79.4 nM T80975 CS6TJ8 127027297 IC50 = 86.74 nM T80975 C0EZA2 127027298 IC50 > 500 nM T80975 CER0Q3 127027305 IC50 = 57.36 nM T80975 CAH9J6 127027306 IC50 > 500 nM T80975 CN3SW5 127027307 IC50 = 86.67 nM T80975 CC0R4L 127027308 IC50 = 106.52 nM T80975 C9E7CQ 127027332 IC50 > 10000 nM T80975 CA59WC 127027333 IC50 > 10000 nM T80975 CQXW85 127027334 IC50 > 10000 nM T80975 CPLE01 127027335 IC50 > 10000 nM T80975 CSM76Y 127027336 IC50 > 10000 nM T80975 C6ZX2Y 127027370 IC50 = 215 nM T80975 CT2YZ6 127027371 IC50 > 10000 nM T80975 CE2LV9 127027372 IC50 > 10000 nM T80975 CCXA80 127027373 IC50 > 10000 nM T80975 C7EYC2 127027620 IC50 = 52.2 nM T80975 C12ODR 127027621 IC50 = 213.48 nM T80975 CA7JW5 127027622 IC50 > 500 nM T80975 CMT3C7 127027623 IC50 = 491.9 nM T80975 C0T3HO 127027641 IC50 = 390.4 nM T80975 CLO6P4 127027642 IC50 = 222.59 nM T80975 CV2AY4 127027714 IC50 = 98 nM T80975 C0Q6RG 127027992 IC50 = 560 nM T80975 CHLF80 127028028 IC50 = 59 nM T80975 CY5OQ9 127028029 IC50 = 153 nM T80975 CZ7C3D 127028030 IC50 = 74 nM T80975 CL0W8U 127028035 IC50 = 865 nM T80975 C7PX3L 127028036 IC50 = 840 nM T80975 C39IBG 127028037 IC50 = 918 nM T80975 CD5I1F 127028038 IC50 = 754 nM T80975 C04MHS 127028310 IC50 = 1810 nM T80975 C85ZEY 127028311 IC50 = 1710 nM T80975 C5V3SU 127028312 IC50 = 1860 nM T80975 C6C0QK 127028313 IC50 = 870 nM T80975 C9XH6D 127028969 IC50 = 2020 nM T80975 C9CMQ6 127028970 IC50 = 4720 nM T80975 CXFB96 127028971 IC50 = 4190 nM T80975 C64UOV 127029263 IC50 = 2000 nM T80975 C1XD6R 127029809 IC50 = 542.6 nM T80975 CI1E5W 127029864 IC50 = 86.25 nM T80975 C0HN2Y 127030123 IC50 > 100000 nM T80975 C7S9GI 127030124 IC50 > 100000 nM T80975 CHGN68 127030424 IC50 = 2060 nM T80975 CRV62L 127030425 IC50 > 100000 nM T80975 CF7JT8 127030426 IC50 > 100000 nM T80975 C5YCU2 127030427 IC50 > 100000 nM T80975 CB3J5F 127030529 IC50 = 1400 nM T80975 C0GES2 127031075 IC50 > 100000 nM T80975 CFJ32Y 127031076 IC50 > 100000 nM T80975 COVM25 127031362 IC50 = 5760 nM T80975 CC8V4J 127031368 IC50 > 100000 nM T80975 C78GYH 127031383 IC50 > 31600 nM T80975 C5WA9Z 127031384 IC50 > 100000 nM T80975 CD7LN1 127031385 IC50 = 1100 nM T80975 CI0VX4 127031386 IC50 = 16000 nM T80975 CO89TC 127031387 IC50 = 1990 nM T80975 C7YRK2 127031656 IC50 = 4670 nM T80975 CAM4S5 127031675 IC50 = 12000 nM T80975 C4QD0M 127031676 IC50 = 17060 nM T80975 C0LTC3 127031677 IC50 > 100000 nM T80975 C2U0HN 127031755 IC50 = 280 nM T80975 CR5M3P 127032029 IC50 = 17 nM T80975 C06SZO 127032238 IC50 = 636 nM T80975 C83CIL 127032326 IC50 > 10000 nM T80975 CO1G2K 127032542 IC50 > 31600 nM T80975 CIZ84M 127032568 IC50 = 5120 nM T80975 C12IOL 127033165 IC50 > 100000 nM T80975 CJ4CM1 127033200 IC50 = 3680 nM T80975 CHGK92 127033201 IC50 = 3870 nM T80975 CS6HB9 127033202 IC50 = 1340 nM T80975 CUOD36 127033203 IC50 = 754 nM T80975 C6HXA1 127033204 IC50 = 3450 nM T80975 CTB20X 127033206 IC50 = 473 nM T80975 CE81GT 127033207 IC50 = 460 nM T80975 CAP2Q3 127033208 IC50 = 381 nM T80975 C3OE4J 127033209 IC50 = 141 nM T80975 CTJ4A2 127033210 IC50 = 118 nM T80975 C49LZH 127033211 IC50 = 114 nM T80975 CFO82K 127033212 IC50 = 86 nM T80975 C41RQL 127033213 IC50 = 83 nM T80975 CG4FA8 127033217 IC50 = 3970 nM T80975 C5Y3TB 127033497 IC50 = 86 nM T80975 CSG9N6 127033539 IC50 = 73 nM T80975 C5RO0L 127033758 IC50 > 100000 nM T80975 CES05I 127033845 IC50 > 10000 nM T80975 CH23IT 127033855 IC50 = 360 nM T80975 CVX2W5 127033856 IC50 = 260 nM T80975 C6SV1L 127034132 IC50 = 4200 nM T80975 CL5KS6 127034133 IC50 = 840 nM T80975 CD04YX 127034308 IC50 > 100000 nM T80975 CY4SV3 127034402 IC50 = 9500 nM T80975 CKS28E 127034802 IC50 = 104 nM T80975 CWRB15 127034986 IC50 = 68.62 nM T80975 CM09WL 127035009 IC50 = 22.16 nM T80975 CDU87A 127035163 IC50 = 355.15 nM T80975 CWF1A8 127035662 IC50 = 4070 nM T80975 CY1HD7 127035663 IC50 = 3840 nM T80975 CEPL09 127036182 IC50 = 285.39 nM T80975 C87BIU 127036183 IC50 > 500 nM T80975 CR0NI6 127036477 IC50 = 291.21 nM T80975 CM17TO 127036596 IC50 = 33.23 nM T80975 C2HXQ0 127036744 IC50 = 4680 nM T80975 C52JBY 127036758 IC50 = 420.15 nM T80975 C72EXH 127036764 IC50 = 93.02 nM T80975 CS2ZF6 127036820 IC50 = 3390 nM T80975 CKDH35 127036821 IC50 = 1560 nM T80975 C9NUK2 127036822 IC50 = 1350 nM T80975 C0UNQ7 127036823 IC50 = 350 nM T80975 C5S7WY 127036957 IC50 = 4540 nM T80975 C07BOP 127036958 IC50 = 4260 nM T80975 C7V2PM 127036987 IC50 = 4290 nM T80975 C5HM8K 127036988 IC50 = 3420 nM T80975 C38WHL 127036989 IC50 = 2250 nM T80975 CYI9J5 127037130 IC50 = 4160 nM T80975 CQ2M5I 127037131 IC50 = 3510 nM T80975 C3G6NW 127037132 IC50 = 3200 nM T80975 C20HAX 127037599 IC50 = 4270 nM T80975 CS2NX4 127037600 IC50 = 3660 nM T80975 CN28YA 127037601 IC50 = 4350 nM T80975 C4Z0AT 127037602 IC50 = 3950 nM T80975 CM1H9E 127037810 IC50 = 19.8 nM T80975 C40ZQT 127037811 IC50 = 26.1 nM T80975 CKX40V 127037812 IC50 = 0.5 nM T80975 CX1KJ8 127037813 IC50 = 1.7 nM T80975 CYZ4D9 127037814 IC50 = 7.2 nM T80975 CQ4TK1 127037815 IC50 = 0.6 nM T80975 CK6H5T 127038133 IC50 = 0.9 nM T80975 CEYL93 127038134 IC50 = 0.9 nM T80975 C6D3RI 127038157 IC50 = 7.6 nM T80975 C93RQT 127038361 IC50 = 8770 nM T80975 CHMT84 127038362 IC50 = 4340 nM T80975 CVU8Z4 127038363 IC50 = 2340 nM T80975 CB73NS 127038364 IC50 = 7560 nM T80975 C0YS4M 127038477 IC50 = 4.9 nM T80975 CMH23X 127038478 IC50 = 5.2 nM T80975 C8BZJ6 127038479 IC50 = 1.8 nM T80975 C70RUP 127038480 IC50 = 0.5 nM T80975 C0PLD4 127038481 IC50 = 2.2 nM T80975 C3FCT9 127038482 IC50 = 2.3 nM T80975 CJHQ62 127038729 IC50 = 2870 nM T80975 CB8XU5 127038848 IC50 = 3.2 nM T80975 CRW80Y 127038849 IC50 = 2.1 nM T80975 C4CUH2 127038850 IC50 = 2.9 nM T80975 C6JSL5 127038851 IC50 = 6 nM T80975 CQ67OE 127038852 IC50 = 3 nM T80975 C9EY0G 127039161 IC50 = 2 nM T80975 CB3DF5 127039162 IC50 = 6.2 nM T80975 C3NR9T 127039163 IC50 = 1.8 nM T80975 C2K4EO 127039164 IC50 = 2.2 nM T80975 CCX3I6 127039165 IC50 = 3.8 nM T80975 CSV0T8 127039237 IC50 = 886 nM T80975 CW4S0U 127039718 IC50 = 3450 nM T80975 C8BSO6 127039719 IC50 = 4360 nM T80975 CNH94T 127039720 IC50 = 2390 nM T80975 C01LGZ 127039804 IC50 = 4490 nM T80975 C3N2YV 127039870 IC50 = 478 nM T80975 C64ZXD 127039985 IC50 = 17 nM T80975 CCG72S 127040317 IC50 = 118 nM T80975 CYB4X0 127041171 IC50 = 19.2 nM T80975 C8TB3R 127041351 IC50 = 3 nM T80975 C40WEH 127041352 IC50 = 0.86 nM T80975 CYM0T6 127041396 IC50 = 3450 nM T80975 CXM5Q6 127041397 IC50 = 4330 nM T80975 CJI9D7 127041398 IC50 = 3490 nM T80975 CGX1C5 127041399 IC50 = 2340 nM T80975 CRY1L6 127041473 IC50 = 2 nM T80975 CH39YG 127041474 IC50 = 1.3 nM T80975 CPE4Z0 127041475 IC50 = 4.1 nM T80975 C05ZWS 127041476 IC50 = 1.3 nM T80975 C0M8RQ 127041477 IC50 = 8.8 nM T80975 C1YC9M 127041601 IC50 = 8 nM T80975 C1S2RM 127041774 IC50 = 3 nM T80975 C0U6IX 127041775 IC50 = 3.7 nM T80975 CUV50M 127041776 IC50 = 2 nM T80975 C3WCN8 127041777 IC50 = 1.2 nM T80975 CC0A1T 127041778 IC50 = 1.4 nM T80975 CZ80JG 127042662 IC50 = 2.1 nM T80975 C1G9QI 127042685 IC50 = 2450 nM T80975 CZ3J4V 127042686 IC50 = 3450 nM T80975 C27XTM 127042687 IC50 = 4560 nM T80975 CYU8Z5 127043892 IC50 = 1030 nM T80975 C9MP2B 127043910 IC50 > 10000 nM T80975 CO6ZX5 127045058 IC50 = 33 nM T80975 C4SFJ8 127045059 IC50 = 450 nM T80975 C08FHU 127045060 IC50 = 3 nM T80975 C8FZV7 127045061 IC50 = 134 nM T80975 CC9MH7 127045070 IC50 = 7100 nM T80975 CAQT96 127045071 IC50 = 1520 nM T80975 C8EVZ2 127045072 IC50 = 5300 nM T80975 C3SMP8 127045121 IC50 = 250 nM T80975 CSF7P8 127045191 IC50 = 10000 nM T80975 C2IP1U 127045218 IC50 > 10000 nM T80975 C0Z8PX 127045223 IC50 = 11 nM T80975 CZL48B 127045224 IC50 = 310 nM T80975 CU2D3X 127045225 IC50 = 21 nM T80975 CSQ06E 127045273 IC50 = 120 nM T80975 CC6W0E 127045274 IC50 = 99 nM T80975 CH6D5S 127045335 IC50 = 2400 nM T80975 C5AXB2 127045351 IC50 = 4400 nM T80975 CY8BX9 127045352 IC50 = 36 nM T80975 CC6WS4 127045353 IC50 = 78 nM T80975 CZ0TP1 127045361 IC50 = 51 nM T80975 CFSX97 127045494 IC50 = 6600 nM T80975 CHK16Q 127045929 IC50 > 1000 nM T80975 CF2U9X 127045946 IC50 = 17.5 nM T80975 CMD1Y6 127046108 IC50 > 10000 nM T80975 CD4G0C 127046310 IC50 > 10000 nM T80975 C5KX9R 127046975 IC50 > 10000 nM T80975 CT0SU2 127046976 IC50 > 10000 nM T80975 CN2ZV4 127047233 IC50 > 100 nM T80975 CL5IA8 127047296 IC50 = 35.8 nM T80975 CGV28E 127047354 IC50 > 100 nM T80975 CY3J0C 127047591 IC50 > 1000 nM T80975 CL8GM6 127047677 IC50 > 10000 nM T80975 CQPV90 127047678 IC50 > 10000 nM T80975 CHTS05 127047813 IC50 > 10000 nM T80975 C6B1MP 127047814 IC50 > 10000 nM T80975 C9SI5T 127047969 IC50 = 21.5 nM T80975 C9F1CL 127048332 IC50 = 890 nM T80975 C2V7JE 127048360 IC50 = 57.9 nM T80975 C9PW5M 127050054 IC50 = 145 nM T80975 CD0K5H 127050299 IC50 = 114 nM T80975 CJU6L2 127050336 IC50 = 24.5 nM T80975 C61QRY 127050340 IC50 = 690 nM T80975 CRYV95 127051004 IC50 = 237 nM T80975 CA91PL 127051005 IC50 = 81 nM T80975 CWM53H 127051274 IC50 = 117 nM T80975 CW9A5D 127051902 IC50 = 201 nM T80975 CG85OA 127051903 IC50 = 168 nM T80975 CA97MR 127052127 IC50 = 220 nM T80975 CA43DP 127052672 IC50 > 5000 nM T80975 C9TQG2 127052673 IC50 = 3000 nM T80975 C0FM1R 130196825 IC50 = 3934 nM T80975 CUO41K 130470684 IC50 = 79000 nM T80975 CT06ZP 132008468 IC50 = 95.3 nM T80975 C96WRI 132008498 IC50 = 20.8 nM T80975 CUO0C5 132156633 IC50 > 10000 nM T80975 CV8DP9 132487332 IC50 = 27.13 nM T80975 CS31LI 132528943 IC50 = 3600 nM T80975 C2AQ0S 132528944 IC50 = 1200 nM T80975 CJ04HZ 132585195 IC50 = 2280 nM T80975 CL6E4J 132601725 IC50 > 25000 nM T80975 CI2YE9 132606873 IC50 = 162.6 nM T80975 C53OJM 132607333 IC50 = 151.52 nM T80975 CMI3Q0 132819888 IC50 = 589 nM T80975 CERS64 132937256 IC50 = 20618 nM T80975 CN9SD7 132942957 IC50 = 67.3 nM T80975 CMP2S9 132942958 IC50 = 13.6 nM T80975 C6CYV4 134132651 IC50 > 10000 nM T80975 C3NEU6 134133052 IC50 = 8.5 nM T80975 C1BTI2 134133235 IC50 = 0.41 nM T80975 C6IU4F 134133491 IC50 = 588 nM T80975 CZT6O0 134133815 IC50 = 0.55 nM T80975 CI53QU 134133842 IC50 = 6.1 nM T80975 CG8M5O 134134176 IC50 = 9.7 nM T80975 CH3QN8 134135021 IC50 = 0.42 nM T80975 C3COF8 134135258 IC50 = 0.54 nM T80975 CR5F3L 134135362 IC50 = 214 nM T80975 CV4Q0M 134135529 IC50 = 404 nM T80975 CEQ1M7 134135734 IC50 = 815 nM T80975 CK9W4F 134135741 IC50 = 2900 nM T80975 CD1O7N 134136322 IC50 > 10000 nM T80975 C3LX0Z 134136666 IC50 = 3.6 nM T80975 CN79XJ 134137614 IC50 = 14 nM T80975 CK15UI 134137837 IC50 = 1986 nM T80975 C45HRS 134139393 IC50 = 576 nM T80975 C5OEI3 134139438 IC50 = 1.2 nM T80975 CJ9RI1 134140064 IC50 = 14 nM T80975 CFAW82 134141290 IC50 = 9.8 nM T80975 C62GWK 134141404 IC50 = 1100 nM T80975 C6HD9W 134141630 IC50 = 5.7 nM T80975 CS95WZ 134142314 IC50 = 966 nM T80975 CP38FT 134142454 IC50 > 10000 nM T80975 C7TF6I 134142952 IC50 = 0.43 nM T80975 CJT12G 134143005 IC50 = 2.7 nM T80975 CMA60G 134144799 IC50 = 2700 nM T80975 C3MN6B 134144868 IC50 = 410 nM T80975 CDMB08 134145603 IC50 > 50000 nM T80975 CB89WK 134145650 IC50 > 10000 nM T80975 CEZH84 134146580 IC50 = 52 nM T80975 CN35SO 134146628 IC50 > 1000 nM T80975 CS7CJ4 134146891 IC50 = 1873 nM T80975 CDF1R9 134147522 IC50 > 10000 nM T80975 C1DF4R 134147544 IC50 = 1600 nM T80975 CS0WH4 134147608 IC50 = 0.77 nM T80975 CUKE45 134147919 IC50 = 480.47 nM T80975 CH5O1F 134148524 IC50 = 178 nM T80975 CFZI08 134149229 IC50 = 18 nM T80975 CU7FX1 134149906 IC50 = 0.69 nM T80975 CIKN06 134150340 IC50 = 0.88 nM T80975 C6CFO5 134150713 IC50 = 79 nM T80975 C76JIM 134151200 IC50 > 10000 nM T80975 CRH2V4 134151618 IC50 = 7.8 nM T80975 C95NCV 134151662 IC50 = 28 nM T80975 C7NB0Z 134152247 IC50 = 275 nM T80975 CG10PO 134152385 IC50 = 7.5 nM T80975 CJ9N1A 134152440 IC50 = 261 nM T80975 C34KQM 134152648 IC50 = 0.67 nM T80975 C8WVZ0 134152967 IC50 = 720 nM T80975 CR09XE 134154074 IC50 = 8.6 nM T80975 C2Q1XW 134154347 IC50 = 2.4 nM T80975 C2ISW7 134155088 IC50 = 279 nM T80975 CR54HK 134155423 IC50 = 528 nM T80975 C29UML 134155621 IC50 = 3200 nM T80975 CX7YE1 134155961 IC50 = 6.5 nM T80975 C2QN7B 134156570 IC50 > 10000 nM T80975 CE38MW 134156584 IC50 = 2.4 nM T80975 CKL8X3 134156658 IC50 = 3.5 nM T80975 CH1GS2 134157091 IC50 = 0.7 nM T80975 CVI25K 134157526 IC50 = 170 nM T80975 CX0UR7 134694318 IC50 > 100000 nM T80975 CYL5V1 134694986 IC50 = 18364 nM T80975 CLCO61 135398510 EC50 = 46 nM T80975 CLSE63 135398512 IC50 = 10 nM T80975 CN5T7W 135400982 IC50 = 210 nM T80975 CVJ07T 135402853 IC50 = 45 nM T80975 C76JPR 135405015 IC50 = 6 nM T80975 CBK6I2 135407156 IC50 = 220 nM T80975 CMVS34 135410282 IC50 = 58 nM T80975 C3K8AZ 135418423 IC50 = 16 nM T80975 CUT52Q 135421574 IC50 = 5800 nM T80975 CT9ZV6 135422893 IC50 = 63 nM T80975 CK9D4A 135428921 IC50 = 380 nM T80975 CV8Q7A 135430397 IC50 = 10 nM T80975 C8X5SV 135433815 IC50 = 240 nM T80975 CUW7X4 135440441 IC50 = 1600 nM T80975 CM4J6A 135444580 IC50 = 34 nM T80975 C2K4QF 135445273 IC50 = 2000 nM T80975 C8GZ2B 135449326 Ki = 3900 nM T80975 CNZ04G 135453357 IC50 = 60 nM T80975 C16XLU 135454992 IC50 = 35 nM T80975 C1M3PW 135458467 IC50 = 16.4 nM T80975 C6U2PZ 135464206 IC50 = 70000 nM T80975 CS63IO 135476717 IC50 = 21 nM T80975 C9D2FL 135483378 IC50 > 4880 nM T80975 CA80OZ 135488014 IC50 = 3 nM T80975 CDCF48 135488027 IC50 = 13 nM T80975 C3IJ9V 135497787 IC50 = 1070 nM T80975 C9YNE7 135497791 IC50 = 640 nM T80975 C8HO5W 135497794 IC50 = 4670 nM T80975 CSP15M 135497800 IC50 = 110 nM T80975 CBF73U 135497834 IC50 > 100 nM T80975 CEKY53 135497841 IC50 > 100 nM T80975 C7GKS9 135497849 IC50 = 150 nM T80975 C3WKV4 135497850 IC50 = 100 nM T80975 CTUB09 135497851 IC50 = 1460 nM T80975 COH6V1 135497852 IC50 = 10000 nM T80975 CU8T6K 135497853 IC50 > 100000 nM T80975 CC58VR 135497854 IC50 = 460 nM T80975 C0ML5X 135497855 IC50 = 1550 nM T80975 C1PJB2 135497865 IC50 = 1000 nM T80975 C1V9AZ 135497869 IC50 = 380 nM T80975 CN2W4U 135497870 IC50 = 10000 nM T80975 C03EJP 135497876 IC50 = 1000 nM T80975 CR09SN 135497877 IC50 = 100 nM T80975 CU6T8C 135497878 IC50 > 100000 nM T80975 C45KEI 135497879 IC50 = 160 nM T80975 C64EMD 135500075 IC50 = 18 nM T80975 CG5HY4 135507297 IC50 < 10 nM T80975 CVZ08D 135509841 IC50 = 600 nM T80975 CK5G2W 135510524 IC50 = 25 nM T80975 CR51FT 135511450 IC50 = 67000 nM T80975 CT0NV5 135514617 IC50 = 22 nM T80975 CTJ48K 135524085 IC50 = 190 nM T80975 CUT1W7 135524168 IC50 = 100 nM T80975 CWHC56 135532320 IC50 = 157 nM T80975 CTW68N 135532699 IC50 = 43 nM T80975 CFPV27 135543821 IC50 = 17 nM T80975 CRCH86 135546221 IC50 = 279 nM T80975 C65XMQ 135546228 IC50 = 4 nM T80975 CTB7R2 135564980 IC50 = 12 nM T80975 CZKG81 135566619 IC50 = 620 nM T80975 C19QOB 135620673 IC50 = 760 nM T80975 C37RUJ 135620674 IC50 = 1700 nM T80975 CD08US 135620675 IC50 = 290 nM T80975 CADG57 135620676 IC50 = 1280 nM T80975 C4XV9S 135620677 IC50 = 650 nM T80975 CO9L3F 135620678 IC50 = 1350 nM T80975 C0IXJ4 135620680 IC50 = 610 nM T80975 C23VIF 135653162 IC50 = 3330 nM T80975 CW08GF 135674125 IC50 = 860 nM T80975 CLS64T 135674129 IC50 = 940 nM T80975 C54ABM 135674133 IC50 = 17 nM T80975 CM7YH4 135674136 IC50 = 66 nM T80975 C1WSO7 135674140 IC50 = 6500 nM T80975 CA0Y7V 135674142 IC50 = 66 nM T80975 CM90FP 135674144 IC50 = 26 nM T80975 C3CP1X 135674147 IC50 = 14 nM T80975 CBSV42 135674149 IC50 = 57 nM T80975 C1NTB0 135674153 IC50 = 42 nM T80975 CID0W9 135674167 IC50 = 5 nM T80975 C1DL9J 135674173 IC50 = 220 nM T80975 CO89UX 135674193 IC50 = 43 nM T80975 CPV59N 135685787 Ki = 3400 nM T80975 CZ49HM 135723775 IC50 = 820 nM T80975 CU29YK 135750268 IC50 = 1450 nM T80975 C6V4DX 135794286 IC50 = 970 nM T80975 CO21NR 135823061 IC50 = 10000 nM T80975 CX4ZB3 135863110 IC50 = 10000 nM T80975 CD5FG3 135867275 IC50 = 650 nM T80975 CE95HA 135922389 IC50 = 3060 nM T80975 C3BZ4A 135922390 IC50 > 10000 nM T80975 C2H3XB 135926086 IC50 = 27 nM T80975 C7BES6 135926087 IC50 = 53 nM T80975 CNTK81 135926088 IC50 = 19 nM T80975 CQ64OH 135926089 IC50 = 980 nM T80975 CXG7O4 135926090 IC50 = 50 nM T80975 CN4FG3 135926091 IC50 = 560 nM T80975 C7NZU3 135926094 IC50 > 25000 nM T80975 CL6HQ4 135926104 IC50 = 29 nM T80975 CE37KQ 135926113 IC50 = 12 nM T80975 C1ZRT7 135926114 IC50 = 78 nM T80975 CU5W2V 135926115 IC50 = 160 nM T80975 C1D3EW 135926116 IC50 = 21 nM T80975 C3YO9W 135929504 IC50 = 2000 nM T80975 C1NH5A 135929506 IC50 > 100000 nM T80975 CA8UN4 135929507 IC50 > 100000 nM T80975 C7J9ZD 135929508 IC50 = 12000 nM T80975 CB2P3H 135929509 IC50 = 630 nM T80975 CJ1S7B 135929510 IC50 = 8600 nM T80975 C4IMU5 135929525 IC50 = 1800 nM T80975 C65NTO 135929526 IC50 = 87000 nM T80975 CAV34T 135929527 IC50 = 16000 nM T80975 C9EX0T 135929541 IC50 = 2700 nM T80975 CE4OU5 135929542 IC50 = 670 nM T80975 C01HMT 135932346 IC50 = 34 nM T80975 CF1PS8 135934877 Ki = 1800 nM T80975 CIPA79 135937899 IC50 = 6900 nM T80975 C12UDA 135947972 IC50 = 1530 nM T80975 CN42ZS 135947973 IC50 = 213 nM T80975 CF8AO3 135947974 IC50 = 8100 nM T80975 CW08GJ 135947976 IC50 = 8100 nM T80975 CJN7E2 135947978 IC50 = 100000 nM T80975 CFKH34 135947979 IC50 = 10 nM T80975 CTRL59 135976660 Ki = 1000 nM T80975 C9UWM5 135980535 IC50 = 1000 nM T80975 CU04CY 135980536 IC50 = 6000 nM T80975 C1XRN3 135980537 IC50 = 5000 nM T80975 CBY03K 135980538 IC50 = 200 nM T80975 C61ZAB 135980539 IC50 = 600 nM T80975 CZC4N6 135980540 IC50 = 1 nM T80975 CLY75R 135980541 IC50 = 200 nM T80975 CYO2Q5 135980542 IC50 = 800 nM T80975 CVRS52 135980544 IC50 = 0.3 nM T80975 CLWH13 135980545 IC50 = 1.3 nM T80975 CU85DF 135980546 IC50 = 4.9 nM T80975 C7BXK1 135980548 IC50 = 300 nM T80975 C8Z6TL 135980550 IC50 = 1100 nM T80975 C4HE8R 135980551 IC50 = 4.3 nM T80975 CH5EF4 135980552 IC50 = 35 nM T80975 C83IKO 135980553 IC50 = 760 nM T80975 CR02QX 135980554 IC50 = 300 nM T80975 CES8N2 135980555 IC50 = 1050 nM T80975 CD3VA2 135980562 IC50 = 300 nM T80975 CM9BS2 135980563 IC50 = 13 nM T80975 C89EHY 135980564 IC50 = 19 nM T80975 C1YS9F 135980565 IC50 = 1100 nM T80975 CN1XQ8 135980566 IC50 = 16 nM T80975 C9GBJ0 135980567 IC50 = 740 nM T80975 CV6E0T 135980569 IC50 = 22 nM T80975 CJ10OI 135980570 IC50 = 280 nM T80975 C2A4BF 135980571 IC50 = 400 nM T80975 C1EN7V 135980572 IC50 = 1.3 nM T80975 CEH8S3 135980573 IC50 = 0.7 nM T80975 C6R5QU 135980574 IC50 = 6.7 nM T80975 C7TL8P 135980575 IC50 = 8 nM T80975 C9MWY0 135980576 IC50 = 8.6 nM T80975 CX9IL5 135980577 IC50 = 0.5 nM T80975 C52VUG 135980579 IC50 = 2.1 nM T80975 CY57BS 135980580 IC50 = 46 nM T80975 C4RL7Q 135985508 IC50 = 480 nM T80975 CXM75Z 135985610 IC50 = 32 nM T80975 C86BZJ 135988997 IC50 = 22 nM T80975 C3IP7O 135995901 IC50 = 5610 nM T80975 CSI70N 135995902 IC50 = 4260 nM T80975 C12OBT 135995903 IC50 = 5090 nM T80975 C3WZ6X 135995904 IC50 = 2580 nM T80975 CARW68 135995905 IC50 = 2510 nM T80975 C3SM2G 135995906 IC50 = 2120 nM T80975 C7UTD0 135995907 IC50 = 1990 nM T80975 CNA78C 135995908 IC50 = 1930 nM T80975 CA56NS 135995909 IC50 = 2670 nM T80975 C5VH7I 135995910 IC50 = 3920 nM T80975 C13VAN 135998871 IC50 = 1312 nM T80975 C1RG8B 135998872 IC50 = 2099 nM T80975 C9W6BT 136002660 IC50 = 39 nM T80975 CD9CT6 136002661 IC50 = 34 nM T80975 C4T9KZ 136002662 IC50 = 33 nM T80975 CU1DK6 136002681 IC50 = 32.7 nM T80975 CJID74 136013449 IC50 = 2600 nM T80975 CHA4N2 136013680 IC50 > 10 nM T80975 C3IDZ7 136043846 IC50 = 500 nM T80975 C13VUJ 136048734 IC50 = 80 nM T80975 C23CNH 136048799 IC50 = 320 nM T80975 C4KUG0 136048800 IC50 = 240 nM T80975 CJ7U4C 136053657 IC50 = 210.2 nM T80975 CAW0E4 136065882 IC50 > 100000 nM T80975 CG1R7B 136087060 IC50 > 10000 nM T80975 C4S6UX 136094844 IC50 = 2700 nM T80975 CS4R2M 136098630 IC50 = 18 nM T80975 CWM2S3 136098631 IC50 = 4760 nM T80975 CFKB53 136104460 IC50 = 29000 nM T80975 C8EBH1 136105653 IC50 = 1080 nM T80975 C4IP6Q 136117936 IC50 = 8 nM T80975 CH1S0I 136117937 IC50 = 174 nM T80975 C7URP5 136117938 IC50 = 35 nM T80975 CDS32V 136117939 IC50 = 28 nM T80975 CL05PS 136117940 IC50 = 10 nM T80975 CFY7U4 136117942 IC50 = 56 nM T80975 C58UOE 136117943 IC50 = 48 nM T80975 CD0VF6 136117946 IC50 = 16 nM T80975 C2LE4F 136117947 IC50 = 110 nM T80975 C9O2EW 136117950 IC50 = 22 nM T80975 CFG58K 136117954 IC50 = 34 nM T80975 CJ8IS3 136117955 IC50 = 73 nM T80975 C9P7AJ 136117956 IC50 = 6 nM T80975 CWJ6N3 136117957 IC50 = 89 nM T80975 C0A2XB 136117958 IC50 = 16 nM T80975 CDY96P 136117961 IC50 = 73 nM T80975 C2BWY4 136117964 IC50 = 12 nM T80975 C6MN3W 136117967 IC50 = 13 nM T80975 CPX4O7 136117969 IC50 = 25 nM T80975 C1Y0PS 136118031 IC50 > 100000 nM T80975 CA76XZ 136118032 IC50 = 100000 nM T80975 CVQ41X 136118033 IC50 > 10000 nM T80975 CU5XR2 136118034 IC50 = 110 nM T80975 C4G6PT 136118035 IC50 = 1600 nM T80975 CU05YS 136118622 IC50 = 145 nM T80975 CN49OS 136118623 IC50 = 128 nM T80975 C39CXW 136118624 IC50 = 157 nM T80975 CR48NF 136118625 IC50 = 1134 nM T80975 CD5M9T 136118626 IC50 = 660 nM T80975 CW27AO 136118641 IC50 = 1950 nM T80975 CZHA29 136118700 IC50 = 97 nM T80975 CFD03R 136118701 IC50 = 119 nM T80975 C3SIK1 136118702 IC50 = 88 nM T80975 C4LC2Q 136118703 IC50 = 633 nM T80975 CX39CA 136118704 IC50 = 125 nM T80975 C3PI2X 136118707 IC50 = 106 nM T80975 C2OAK8 136118708 IC50 = 290 nM T80975 C6PUG0 136118709 IC50 = 19903 nM T80975 CH1E7I 136118710 IC50 = 2180 nM T80975 C0RBJ7 136118711 IC50 = 327 nM T80975 C4V8HY 136118712 IC50 = 9876 nM T80975 CZ4AF8 136118717 IC50 = 68 nM T80975 CMP78A 136118718 IC50 = 51 nM T80975 CN8RB4 136118719 IC50 = 4880 nM T80975 CIUJ95 136118720 IC50 = 4880 nM T80975 C2BIZ5 136118721 IC50 = 4 nM T80975 C5YL7I 136118722 IC50 = 213 nM T80975 CZQ5P1 136118733 IC50 = 23633 nM T80975 CMP4R8 136118734 IC50 = 5 nM T80975 C7E6XJ 136118735 IC50 = 82 nM T80975 CCX81R 136118736 IC50 = 3 nM T80975 C29ZXF 136118737 IC50 = 60 nM T80975 C5QZ4H 136126664 IC50 > 25000 nM T80975 CB8RX0 136126665 IC50 = 170 nM T80975 CQ84IZ 136180335 Ki > 4000 nM T80975 CZ7EX0 136183413 IC50 = 310 nM T80975 CC52HL 136189674 IC50 > 3600 nM T80975 C6HW4E 136206295 IC50 = 9200 nM T80975 CU9P3M 136206296 IC50 = 7500 nM T80975 C2OQ8Z 136211076 IC50 = 9 nM T80975 CDT7E4 136211077 IC50 = 7.5 nM T80975 C9RE8D 136215817 IC50 = 384.1 nM T80975 C1YUD0 136219394 IC50 > 10 nM T80975 C5TQJ3 136227998 IC50 = 2250 nM T80975 C5S3WN 136228008 IC50 = 15300 nM T80975 CKHE36 136254163 IC50 = 600 nM T80975 CIU8W3 136254389 IC50 > 10 nM T80975 CE7L0G 136269119 IC50 > 50000 nM T80975 C7U9GP 136269138 IC50 > 50000 nM T80975 CF3BX6 136269606 IC50 = 78 nM T80975 CM5E6A 136269610 IC50 = 45 nM T80975 CK7AX4 136269611 IC50 = 42 nM T80975 CK5JF1 136269612 IC50 = 12 nM T80975 C35MBU 136299423 IC50 = 12 nM T80975 C0W8KA 136299435 IC50 = 1.6 nM T80975 C5G4ES 136299436 IC50 = 8.3 nM T80975 CE8BT2 136347029 IC50 = 32000 nM T80975 CFQO70 136375226 IC50 = 630 nM T80975 CC8Q2D 136375233 IC50 = 2500 nM T80975 CJD5N7 136986961 IC50 = 12 nM T80975 C9H4GB 136998821 IC50 = 9530 nM T80975 C9Z2YQ 137028533 IC50 = 40100 nM T80975 C0Y3EV 137028534 IC50 = 6960 nM T80975 CQ02OI 137062185 IC50 = 750 nM T80975 C4FB9U 137062186 IC50 = 710 nM T80975 CUW85H 137062187 IC50 = 310 nM T80975 CW0FE9 137083622 IC50 > 10000 nM T80975 CL4M3P 137133110 IC50 = 12.6 nM T80975 CNUX28 137133111 IC50 = 2.5 nM T80975 CXR23D 137133115 IC50 = 8 nM T80975 CL2I8P 137133138 IC50 = 7.8 nM T80975 C83WAK 137189946 IC50 = 3450 nM T80975 C8KW0I 137189951 IC50 = 3220 nM T80975 COX23B 137189952 IC50 = 3450 nM T80975 CCM42D 137249694 IC50 = 51.7 nM T80975 CXT8B9 137287443 IC50 = 4.4 nM T80975 CE75QD 137321162 IC50 = 850 nM T80975 CM4TU2 137321167 IC50 > 1000 nM T80975 CCX3Q6 137628632 IC50 > 10000 nM T80975 C25ERN 137631967 IC50 = 0.8 nM T80975 CORJ86 137632190 EC50 = 3 nM T80975 C9UW0D 137632355 IC50 = 1.05 nM T80975 CV49KX 137632804 IC50 = 1921 nM T80975 CQ7MZ6 137633392 IC50 = 11.41 nM T80975 CE1B7Y 137633677 IC50 = 6228 nM T80975 CS7PJ6 137633789 IC50 > 10000 nM T80975 CFUY16 137633842 IC50 = 10200 nM T80975 CMY81W 137633944 IC50 = 3695 nM T80975 CHC70D 137634143 IC50 = 671.8 nM T80975 CI1E8V 137634241 IC50 = 3350 nM T80975 CPFH76 137634323 IC50 = 11382 nM T80975 C85WBP 137634338 IC50 = 420 nM T80975 CSQ87K 137634450 IC50 = 32.37 nM T80975 CAD3C5 137634686 IC50 = 137.51 nM T80975 CMOK58 137634923 IC50 = 59.9 nM T80975 CKH35C 137635255 Ki = 11070 nM T80975 CILC91 137635352 IC50 = 6920 nM T80975 CS23KQ 137635618 IC50 = 160300 nM T80975 CY4M7O 137635632 Ki = 4470 nM T80975 CBP52G 137635849 IC50 = 3360 nM T80975 C5JD9N 137635898 IC50 = 33 nM T80975 CK5Y3P 137635915 IC50 = 96.22 nM T80975 CK8G2R 137636007 IC50 > 50000 nM T80975 C5T0YN 137636330 EC50 = 47 nM T80975 CEL8G1 137636465 IC50 > 50000 nM T80975 C9F5GA 137636582 IC50 = 0.31 nM T80975 CL1Q8V 137637006 IC50 = 4322 nM T80975 C06JRX 137637094 IC50 = 1.7 nM T80975 C5LU2S 137637274 Ki = 3240 nM T80975 CLFR07 137637309 IC50 = 4164 nM T80975 C4KPZ9 137638346 IC50 = 1.88 nM T80975 CU24QC 137638448 IC50 = 38.7 nM T80975 C6ESL5 137638961 IC50 > 1000 nM T80975 CP2B8Y 137639044 IC50 > 50000 nM T80975 CI7WH5 137639132 IC50 = 1791 nM T80975 CO9D4W 137639407 IC50 = 164.62 nM T80975 C3UBE2 137639638 IC50 = 84.3 nM T80975 CE96AL 137639657 IC50 = 18700 nM T80975 CX95WZ 137639923 IC50 = 7.8 nM T80975 CI5K8B 137640242 IC50 > 50000 nM T80975 C6LE5P 137640904 Ki = 13410 nM T80975 C8TMV6 137641055 IC50 = 0.92 nM T80975 CA70ZG 137641063 IC50 = 41966 nM T80975 CW3C1G 137641107 IC50 = 1208 nM T80975 CBGR42 137641572 IC50 > 1000 nM T80975 CO18WK 137641971 IC50 = 6229 nM T80975 COH24B 137642226 IC50 = 23 nM T80975 C52EZY 137642247 IC50 = 6235 nM T80975 CGEC59 137642439 IC50 = 104.5 nM T80975 CP5Q4H 137642451 IC50 = 34.67 nM T80975 CWB74C 137642729 IC50 = 33.02 nM T80975 CR7DU4 137642765 Ki = 1930 nM T80975 CJ4S0F 137642960 IC50 = 3940 nM T80975 CU8YX6 137643005 IC50 = 193100 nM T80975 CPE93W 137643241 IC50 = 1.42 nM T80975 CVF3Y4 137643942 IC50 = 5613 nM T80975 C2T6FV 137644825 IC50 = 167.51 nM T80975 C9F6VM 137645016 IC50 > 50000 nM T80975 CAY1L6 137645294 IC50 > 1000 nM T80975 CKP7N9 137645385 Ki = 3990 nM T80975 C2BP8R 137645569 IC50 = 4920 nM T80975 C6DOB5 137645672 IC50 > 1000 nM T80975 C9ERJ2 137645774 IC50 = 19 nM T80975 CF92BJ 137646079 IC50 = 26163 nM T80975 CPI1C6 137646147 IC50 > 1000 nM T80975 CN5R6A 137646618 IC50 > 1000 nM T80975 CAL48N 137646892 IC50 = 24 nM T80975 CVZ85B 137647227 IC50 = 700.53 nM T80975 CU5B3H 137647479 IC50 = 15.29 nM T80975 C5B7PN 137647552 IC50 = 9046 nM T80975 C0E5LD 137647791 IC50 > 50000 nM T80975 CITB67 137647879 IC50 > 50000 nM T80975 C8CYG9 137648008 IC50 = 2391 nM T80975 CHKS97 137648071 Ki = 3260 nM T80975 CGI1F8 137649216 IC50 = 10917 nM T80975 CY6UG1 137649571 IC50 = 28.79 nM T80975 CTF9N6 137649662 IC50 = 10462 nM T80975 C08HAC 137649959 IC50 = 3937 nM T80975 C8EQA5 137650407 IC50 = 33.36 nM T80975 C5R6KV 137650589 IC50 = 2.5 nM T80975 CVK6O2 137650604 IC50 > 50000 nM T80975 CI6X0A 137651311 IC50 = 3145 nM T80975 CIM42E 137651341 IC50 = 4293 nM T80975 C1DK0P 137651391 IC50 = 2.6 nM T80975 C5F3LP 137651946 IC50 = 38 nM T80975 CL2GW4 137652151 IC50 = 3503 nM T80975 CQUY83 137652218 IC50 > 500000 nM T80975 CYH05X 137652479 IC50 = 1.35 nM T80975 CJ39LQ 137652784 EC50 = 80 nM T80975 C3LAD6 137652990 IC50 > 100000 nM T80975 CHP3E8 137653224 IC50 = 4079 nM T80975 CZS0M4 137653919 IC50 = 1845 nM T80975 C19AQU 137654195 IC50 = 35.75 nM T80975 C78DVY 137654650 IC50 = 1856 nM T80975 CS21QO 137654848 IC50 > 50000 nM T80975 CIS4O3 137655297 IC50 = 4050 nM T80975 C9ZIV1 137655363 IC50 = 5352 nM T80975 CCXH57 137655416 Ki = 4830 nM T80975 C9JT1N 137655519 IC50 = 182200 nM T80975 C9TEU1 137655771 IC50 = 152.71 nM T80975 CQ70VE 137655849 IC50 > 50000 nM T80975 C4OL7J 137656236 Ki = 7240 nM T80975 C3OP5Q 137656266 IC50 = 8.7 nM T80975 C0RQB3 137656341 IC50 = 4523 nM T80975 CZ4C1M 137656917 IC50 = 3109 nM T80975 CO61JG 137657076 IC50 = 5002 nM T80975 CKVO51 137657233 IC50 = 32.9 nM T80975 C1Q7UO 137657235 IC50 = 5.58 nM T80975 CV9H6B 137657843 IC50 = 15935 nM T80975 CV5H3Z 137657932 IC50 = 3.7 nM T80975 C98AVI 137657952 IC50 > 50000 nM T80975 C2M6IZ 137657987 IC50 > 1000 nM T80975 CPV1S9 137658287 IC50 = 55 nM T80975 C2VRD0 137658292 IC50 > 1000 nM T80975 C81LTC 137658404 IC50 = 6235 nM T80975 CQMB10 137658515 IC50 = 1225 nM T80975 C7IVT9 137658762 IC50 > 200 nM T80975 C8E4QA 137658885 IC50 = 1.4 nM T80975 CX53JP 137658925 IC50 = 8634 nM T80975 C4FKX3 137659066 IC50 = 6816 nM T80975 C0DC5L 137659278 Ki = 4150 nM T80975 C07ACR 137659526 IC50 = 0.75 nM T80975 CKVS16 137659546 IC50 > 50000 nM T80975 CC7L3S 137660340 IC50 = 17.85 nM T80975 C07JTH 137660356 Ki = 850 nM T80975 C8D9NE 137660511 IC50 = 1224 nM T80975 CM5T3L 137660584 IC50 > 50000 nM T80975 C7FZA8 137660733 IC50 = 36890 nM T80975 CQE9M4 137661156 IC50 = 164.54 nM T80975 C8WZ2V 137661264 IC50 = 8008 nM T80975 CM0N3T 137661420 IC50 = 26.7 nM T80975 CZT18Q 137661519 IC50 > 1000 nM T80975 C09NZL 137661683 IC50 = 9760 nM T80975 CHB9P7 137661707 IC50 = 3857 nM T80975 CT43IF 137661858 IC50 = 27.3 nM T80975 CIWG23 138393067 IC50 = 37 nM T80975 C5LQU9 138479230 IC50 = 46.4 nM T80975 CSRI06 138547901 IC50 > 1000 nM T80975 CUXO19 138617501 IC50 = 113.4 nM T80975 CW1XQ6 139188711 IC50 = 290 nM T80975 COB9P2 141456067 IC50 = 560 nM T80975 C7C5TV 141462248 IC50 = 548.4 nM T80975 CSYV02 141488087 IC50 = 357.2 nM T80975 CX50BU 141498081 IC50 = 114 nM T80975 C5FX0T 141498082 IC50 = 125 nM T80975 CEKG27 141498083 IC50 = 79 nM T80975 C75HGY 141498092 IC50 = 110 nM T80975 CTR7D4 141535114 IC50 = 169.9 nM T80975 CO9P7G 145351804 IC50 = 2.9 nM T80975 CNU4M3 145704714 IC50 = 7940 nM T80975 C6VB3O 145925651 IC50 >= 5000 nM T80975 C29XUO 145945978 IC50 > 1000 nM T80975 C6Y5NP 145949388 IC50 > 500 nM T80975 C4HB8M 145949394 IC50 = 21 nM T80975 CB3Z1W 145949428 IC50 = 2.35 nM T80975 CCM27G 145949662 IC50 = 808.5 nM T80975 CVJS01 145949677 IC50 = 9.3 nM T80975 CYEK37 145949698 IC50 > 500 nM T80975 CGB21E 145949773 IC50 > 500 nM T80975 CWQA26 145949916 IC50 = 431.2 nM T80975 CC3S9Y 145949933 IC50 = 111.5 nM T80975 CVTZ73 145950013 IC50 = 108.08 nM T80975 C3Q1CR 145950413 IC50 > 500 nM T80975 CT25FH 145950796 IC50 = 1000 nM T80975 CYF32C 145950953 IC50 = 100 nM T80975 CEM48X 145951001 IC50 = 1410 nM T80975 CRXJ25 145951211 IC50 = 300 nM T80975 C9SOT5 145951403 IC50 = 1260 nM T80975 CKU2J6 145951459 IC50 = 28.95 nM T80975 CO0KI7 145951584 IC50 > 500 nM T80975 C1L2BO 145951639 IC50 = 140 nM T80975 CBL7G4 145951848 IC50 = 424 nM T80975 CWUM46 145952127 IC50 > 500 nM T80975 CHKS76 145952159 IC50 = 63.2 nM T80975 CS5FN6 145952182 IC50 = 122.81 nM T80975 CL1J3N 145952225 IC50 = 7.97 nM T80975 C0U2SX 145952427 IC50 = 415.21 nM T80975 C1G0PH 145952494 IC50 = 41.7 nM T80975 CR9LH4 145952520 IC50 = 106.1 nM T80975 C1C2KL 145952546 IC50 = 11.19 nM T80975 C1KX3F 145952675 IC50 = 21.37 nM T80975 CWU7J4 145952685 IC50 > 500 nM T80975 CY3M1A 145952761 IC50 > 500 nM T80975 CETX79 145953187 IC50 > 500 nM T80975 CQO92P 145953233 IC50 = 7.94 nM T80975 C60XZR 145953297 IC50 = 230 nM T80975 CSLC73 145953358 IC50 = 81.3 nM T80975 CAL30B 145953560 IC50 = 65 nM T80975 C6WB5A 145953633 IC50 > 500 nM T80975 C09BOY 145953698 IC50 > 500 nM T80975 C8K3IT 145953806 IC50 > 500 nM T80975 C0V8SM 145954139 IC50 = 110 nM T80975 CN59EV 145954386 IC50 > 500 nM T80975 CX94IY 145954428 IC50 = 325.82 nM T80975 C9WYS2 145954493 IC50 = 29.9 nM T80975 C5Z3NW 145954580 IC50 = 19.97 nM T80975 CF1T9Y 145954667 IC50 = 77.9 nM T80975 CX80ZF 145954847 IC50 = 17.1 nM T80975 CHBA54 145954987 IC50 > 500 nM T80975 C4CQI1 145955346 IC50 > 500 nM T80975 CFZ39K 145955409 IC50 = 138.3 nM T80975 CFC1R5 145955514 IC50 > 500 nM T80975 CDRQ06 145955547 IC50 = 384.7 nM T80975 C8VN1Y 145955561 IC50 = 34 nM T80975 C2O9XD 145955651 IC50 > 1000 nM T80975 C8YLB0 145955872 IC50 = 18 nM T80975 CBR2Q7 145956253 IC50 = 150.2 nM T80975 C1IX5N 145956333 IC50 = 69.1 nM T80975 C6ZNJ1 145956488 IC50 = 8 nM T80975 CLZH04 145956490 IC50 = 104.6 nM T80975 CZ1X4T 145956589 IC50 = 310.64 nM T80975 CNDL29 145956614 IC50 = 73.4 nM T80975 C1Z5BV 145956656 IC50 > 500 nM T80975 C9GN1B 145956669 IC50 = 90.5 nM T80975 C5VSC7 145956704 IC50 = 3.45 nM T80975 C0Y2TV 145956729 IC50 > 500 nM T80975 CY69RH 145956768 IC50 = 646.5 nM T80975 CJ4F8V 145956840 IC50 = 11.9 nM T80975 CPG5X6 145957058 IC50 = 34.68 nM T80975 CB74GR 145957221 IC50 = 300 nM T80975 CA72LX 145957228 IC50 > 500 nM T80975 CY54UC 145957309 IC50 = 94.62 nM T80975 C7YBO3 145957370 IC50 > 500 nM T80975 CZ6O9G 145957666 IC50 = 7.05 nM T80975 CB4P3U 145957792 IC50 > 500 nM T80975 CMSE06 145957839 IC50 = 19.2 nM T80975 CB1MI9 145957910 IC50 = 4 nM T80975 CS47UF 145958497 IC50 = 51 nM T80975 CY3SV6 145959075 IC50 = 640 nM T80975 CEWQ79 145959077 IC50 = 564000 nM T80975 CZ3G0H 145959478 IC50 = 120.4 nM T80975 CZM5L3 145959497 IC50 = 125.32 nM T80975 CVZ4Q2 145959877 IC50 = 297.02 nM T80975 C7RQ8I 145960033 IC50 = 49.8 nM T80975 CH3YK9 145960253 IC50 > 500 nM T80975 CA9LY3 145960784 IC50 > 500 nM T80975 CRVO52 145960991 IC50 > 1000 nM T80975 C1U6NF 145961006 IC50 > 500 nM T80975 CMZN84 145961642 IC50 > 500 nM T80975 CV4M1Z 145961849 IC50 > 1000 nM T80975 CJT41L 145962084 IC50 = 2400 nM T80975 CCK21X 145962292 IC50 = 31.4 nM T80975 CY7B2V 145962703 IC50 = 40.37 nM T80975 CR75NT 145963742 IC50 = 6.17 nM T80975 C9PKU6 145963750 IC50 = 4.6 nM T80975 C2CMR3 145963883 IC50 = 81 nM T80975 CS2NR4 145964261 IC50 = 1830.3 nM T80975 C65YWX 145964882 IC50 = 1900 nM T80975 CHC3T0 145965031 IC50 > 10000 nM T80975 CP92ZF 145965329 IC50 = 690 nM T80975 CPF3U9 145965371 IC50 = 54 nM T80975 C4NP2V 145965631 IC50 > 50000 nM T80975 C9Y7DO 145965819 IC50 = 136.6 nM T80975 CMI61S 145965843 IC50 = 74 nM T80975 CI9R2E 145966320 IC50 = 83 nM T80975 C9HXI4 145966620 IC50 > 10000 nM T80975 C9H4TP 145966705 IC50 = 11000 nM T80975 CTUF34 145966712 IC50 = 46 nM T80975 CQE9M5 145966810 IC50 = 400 nM T80975 C1EH6C 145967078 IC50 = 7500 nM T80975 CDW83M 145967332 IC50 = 62.5 nM T80975 CR6O2S 145967668 IC50 > 10000 nM T80975 C49QZE 145967671 IC50 = 887 nM T80975 C0UZ6Q 145967831 IC50 = 8663 nM T80975 C2CHJ9 145967839 IC50 > 10000 nM T80975 C8QEZ7 145967870 IC50 = 133 nM T80975 CJO79P 145968146 IC50 = 151.5 nM T80975 C1SIC0 145968151 IC50 = 57 nM T80975 C5E8ZK 145968310 IC50 = 46 nM T80975 CTX9I2 145968517 IC50 = 61 nM T80975 C0Y1IT 145968532 IC50 = 6915 nM T80975 CL0BO5 145968619 IC50 > 10000 nM T80975 CHAU61 145968737 IC50 = 84 nM T80975 CKQ74H 145968788 IC50 = 33 nM T80975 CK1N7F 145968871 IC50 = 508 nM T80975 CBJ0F1 145968889 IC50 > 10000 nM T80975 C0BG4F 145968971 IC50 = 3864 nM T80975 CWJ12M 145969155 IC50 = 66 nM T80975 CP8S3O 145969482 IC50 = 37 nM T80975 CU4OP2 145969694 IC50 = 210 nM T80975 CGW5S1 145969844 IC50 = 7600 nM T80975 CFC48X 145969905 IC50 = 5986 nM T80975 C8WIB7 145969935 IC50 = 277 nM T80975 CB8R3A 145970271 IC50 > 10000 nM T80975 COJ7H5 145970527 IC50 = 8 nM T80975 C2O9EN 145970583 IC50 = 220 nM T80975 C4D3BL 145970607 IC50 = 74 nM T80975 C8NK3O 145970839 IC50 = 63 nM T80975 CON74U 145970883 IC50 = 133.2 nM T80975 CNDL79 145970990 IC50 = 10.2 nM T80975 CP6QH1 145971042 IC50 > 10000 nM T80975 CMS6P5 145971054 IC50 = 37 nM T80975 CM2QK5 145971454 IC50 > 1000 nM T80975 C8YM3U 145971698 IC50 > 500 nM T80975 CBI6C0 145971699 IC50 = 7.66 nM T80975 CNVT54 145971746 IC50 = 257.2 nM T80975 CAR6T3 145971936 IC50 = 24.33 nM T80975 COX74G 145971999 IC50 = 134.5 nM T80975 CJD5Q1 145972024 IC50 = 91.7 nM T80975 CDB5N6 145972176 IC50 = 2.1 nM T80975 C3Q4XM 145972183 IC50 = 4.9 nM T80975 C8S6VJ 145972201 IC50 > 500 nM T80975 CO5Z4B 145972302 IC50 > 1000 nM T80975 CG8R0P 145972697 IC50 = 1.9 nM T80975 CZ5P0E 145972710 IC50 > 500 nM T80975 C40VIL 145972979 IC50 = 4500 nM T80975 C87WHG 145973554 IC50 = 44 nM T80975 CLN2D9 145973734 IC50 = 2700 nM T80975 CQBY19 145974023 IC50 = 7700 nM T80975 CXRY95 145974888 IC50 = 450 nM T80975 C74TYP 145975351 IC50 = 291.3 nM T80975 CM7K0A 145975625 IC50 = 48 nM T80975 CF59KI 145976265 IC50 = 20.6 nM T80975 C76RQZ 145976309 IC50 = 2000 nM T80975 CZB63Y 145976371 IC50 = 5.9 nM T80975 CBR8K6 145976838 IC50 = 2300 nM T80975 C59VIT 145977243 IC50 > 50000 nM T80975 C4X7CT 145977420 IC50 > 10000 nM T80975 C93ZOX 145977611 IC50 = 110 nM T80975 CLA57T 145978300 IC50 > 10000 nM T80975 C9DE2V 145979557 IC50 = 101.6 nM T80975 C5TP2U 145979643 IC50 = 14400 nM T80975 CX63VM 145980115 IC50 = 83.7 nM T80975 CNS6I5 145980673 IC50 = 209.3 nM T80975 CR0JD7 145981097 IC50 = 329.5 nM T80975 CR39TX 145981127 IC50 = 6.6 nM T80975 CK96JF 145981325 IC50 = 5 nM T80975 CU25SM 145981644 IC50 = 8.3 nM T80975 CAK6O4 145981649 IC50 = 200 nM T80975 C5YCJ0 145982003 IC50 = 21.6 nM T80975 CQ8A6B 145982177 IC50 = 30 nM T80975 CCS92I 145982511 IC50 = 167 nM T80975 C7UH4A 145982555 IC50 > 1000 nM T80975 C9KR5H 145982571 IC50 > 1000 nM T80975 CWE21T 145982588 IC50 = 105 nM T80975 CC12YA 145982666 IC50 = 12.7 nM T80975 C8UZV2 145982754 IC50 > 1000 nM T80975 CF4BO8 145982785 IC50 = 7.8 nM T80975 CM6ZS7 145982824 IC50 = 15.6 nM T80975 CABC08 145982974 IC50 = 270 nM T80975 C0O1NY 145983278 IC50 > 1000 nM T80975 CF28AU 145983389 IC50 = 23.4 nM T80975 CRL19G 145983447 IC50 = 25 nM T80975 CXB4L8 145983465 IC50 > 1000 nM T80975 C48UZH 145983504 IC50 = 259 nM T80975 C8BZC5 145983753 IC50 = 11 nM T80975 CD5L8O 145983778 IC50 > 200 nM T80975 CQ6XL2 145983816 IC50 = 67 nM T80975 C45JGB 145983851 IC50 = 620 nM T80975 C2WH1T 145983975 IC50 > 1000 nM T80975 C2SMN0 145983991 IC50 = 110 nM T80975 C1YQ8U 145984124 IC50 > 1000 nM T80975 CVH6Y9 145984234 IC50 > 1000 nM T80975 C4C2OM 145984258 IC50 = 3 nM T80975 C9DHL3 145984282 IC50 = 696 nM T80975 C0N4GL 145984412 IC50 > 1000 nM T80975 CU02KG 145984478 IC50 > 1000 nM T80975 CRV38J 145984530 IC50 > 1000 nM T80975 CVT02P 145984555 IC50 = 177 nM T80975 CHW8E5 145984671 IC50 = 130 nM T80975 CQ9A0N 145984791 IC50 = 174 nM T80975 CYG42V 145984818 IC50 > 200 nM T80975 CFS7D5 145984941 IC50 > 200 nM T80975 C05IMJ 145984942 IC50 = 12 nM T80975 CA6L7I 145985051 IC50 > 1000 nM T80975 CEF7W4 145985090 IC50 = 85 nM T80975 C5WVP1 145985325 IC50 = 203 nM T80975 CLGE45 145985395 IC50 = 12 nM T80975 CC3U1S 145985468 IC50 > 1000 nM T80975 CW49HX 145985540 IC50 > 1000 nM T80975 CV96GO 145985569 IC50 = 730 nM T80975 C9Q5VI 145985608 IC50 = 600 nM T80975 CI7G4P 145985681 IC50 = 1600 nM T80975 CA2TW8 145985737 IC50 = 685 nM T80975 CX31WG 145985802 IC50 > 1000 nM T80975 CL1ZN2 145985942 IC50 = 101 nM T80975 CS9C8J 145986155 IC50 > 200 nM T80975 CV19MQ 145986257 IC50 > 1000 nM T80975 C9WDL3 145986316 IC50 = 30.3 nM T80975 C03PYD 145986466 IC50 < 1000 nM T80975 CN9RZ4 145986531 IC50 = 870 nM T80975 C10TUA 145986573 IC50 = 4016 nM T80975 C1Y5MO 145987062 IC50 = 152.3 nM T80975 CH7I9T 145987129 IC50 = 1970 nM T80975 CV75AR 145987208 IC50 = 4.1 nM T80975 CM3FP6 145987671 IC50 = 7.2 nM T80975 C7LV2F 145987970 IC50 = 24.7 nM T80975 C8XD0B 145988239 IC50 = 140.9 nM T80975 CK8S4V 145988419 IC50 = 102 nM T80975 C5EZ1P 145989138 IC50 = 429.8 nM T80975 C0GNE7 145989369 IC50 = 198.5 nM T80975 CT9D0X 145989541 IC50 = 317.6 nM T80975 C2B0LS 145989721 IC50 = 237.3 nM T80975 CI3B9F 145989892 IC50 = 205.2 nM T80975 CACF81 145990005 IC50 = 1200 nM T80975 CJS9Z0 145990229 IC50 = 16 nM T80975 CFM97W 145990241 IC50 = 110.1 nM T80975 C58ODP 145991046 IC50 = 12.4 nM T80975 C3LB2R 145991081 IC50 = 6.1 nM T80975 CLK61X 145992276 IC50 = 12.2 nM T80975 CSKU38 145992346 IC50 = 1220 nM T80975 CNC69T 145992844 IC50 = 8900 nM T80975 CAK5V0 145992869 IC50 = 84.5 nM T80975 C0YA9U 145993477 IC50 = 697.3 nM T80975 CS3DY6 145993716 IC50 = 156.6 nM T80975 C7ER4V 145993972 IC50 = 530 nM T80975 CE4FH2 146018674 IC50 = 9000 nM T80975 C30LIE 146403681 IC50 = 1 nM T80975 CA0ZY2 146403682 IC50 = 1.5 nM T80975 C8ZY5S 146403684 IC50 = 4.2 nM T80975 C5UGO8 146403697 IC50 = 3.4 nM T80975 CX9G0C 146403701 IC50 = 11.2 nM T80975 CG95FV 146403716 IC50 = 2.4 nM T80975 C8SJV4 146403722 IC50 = 4 nM T80975 CI06AK 146403743 IC50 = 31 nM T80975 CZ25RN 146403770 IC50 = 1.5 nM T80975 CST47O 146403779 IC50 = 2.4 nM T80975 C2BH4A 146403800 IC50 = 1.7 nM T80975 C6JCI0 146421555 IC50 = 1081 nM T80975 CBM7C5 146773032 IC50 = 2880 nM T80975 C9D1EH 147117461 IC50 = 3710 nM T80975 C8I1HV 147384518 IC50 = 7160 nM T80975 CC1F9L 147598461 IC50 > 1000 nM T80975 C7DYK4 147709549 IC50 = 6850 nM T80975 CIT79C 148291912 IC50 = 580 nM T80975 C2U0SJ 148390225 IC50 = 10420 nM T80975 CJ23ZE 148637488 IC50 = 3260 nM T80975 CVL49H 149513019 IC50 = 9220 nM T80975 CS8BJ7 149949125 IC50 > 1000 nM T80975 CJL17Q 150336955 IC50 > 1000 nM T80975 C6PG4T 150482255 IC50 > 1000 nM T80975 CP9JW5 150533442 IC50 = 4.15 nM T80975 CHXZ94 151105657 IC50 = 500.28 nM T80975 CU7T8Y 151363744 IC50 = 125.06 nM T80975 C90NHE 151428103 IC50 = 58.1 nM T80975 CFE6I9 152015157 IC50 > 1000 nM T80975 C24QHN 152058632 IC50 = 0.53 nM T80975 CJ4G3V 152221091 IC50 = 0.57 nM T80975 CJSM72 152346156 IC50 = 1.63 nM T80975 CZ7GT5 152346369 IC50 = 3.17 nM T80975 CFKU39 152790957 IC50 = 17350 nM T80975 CV41DF 153011787 IC50 = 10140 nM T80975 CRE82P 155510352 IC50 = 2.57 nM T80975 CF8B4I 155511031 IC50 = 4540 nM T80975 C5Z7GK 155511049 IC50 = 216.77 nM T80975 CFBO36 155511066 IC50 = 1430 nM T80975 CEF6A7 155511067 IC50 = 8.8 nM T80975 C47GVB 155511749 IC50 = 319 nM T80975 CT2U3S 155512176 IC50 = 3980 nM T80975 C18SDP 155512247 IC50 = 2500 nM T80975 C0ZAN6 155512322 IC50 = 250 nM T80975 CL4B2M 155512535 IC50 = 87 nM T80975 CN54EL 155512780 IC50 = 362.7 nM T80975 C7X3WN 155513030 IC50 > 10000 nM T80975 C81YCJ 155513061 IC50 = 94 nM T80975 CQA9U6 155513155 IC50 = 23.1 nM T80975 C2MD1Q 155513187 IC50 > 10000 nM T80975 CCD3B2 155513330 IC50 = 772 nM T80975 CLQ43U 155513345 IC50 = 570 nM T80975 CU12GD 155513666 IC50 = 2390 nM T80975 CC1D3I 155513733 IC50 = 3420 nM T80975 C1XNV5 155513991 IC50 = 3.6 nM T80975 C3VEX4 155514011 IC50 = 2980 nM T80975 C27WHB 155514567 IC50 = 338.3 nM T80975 CMC6N4 155514619 IC50 = 1084 nM T80975 C5K1UD 155514779 IC50 > 1000 nM T80975 C7O1BV 155515046 IC50 = 560 nM T80975 C83CSB 155515100 IC50 = 1.85 nM T80975 C89BUP 155515156 IC50 = 165.9 nM T80975 C8C6YN 155515275 IC50 > 10000 nM T80975 CJ16EX 155516207 IC50 = 4320 nM T80975 CU76NE 155516227 IC50 = 16230 nM T80975 C8XHM5 155516263 IC50 = 17.3 nM T80975 C1S7AI 155516436 IC50 > 1000 nM T80975 C2WRO5 155516460 IC50 = 26.9 nM T80975 CK3Y4E 155516880 IC50 = 113 nM T80975 C73WVL 155517777 IC50 = 46 nM T80975 CPJ4B8 155518090 IC50 = 647 nM T80975 CKH3S7 155518300 IC50 = 256 nM T80975 C86HPW 155518524 IC50 = 31000 nM T80975 C98MWS 155518832 IC50 = 668.7 nM T80975 C3VTM7 155519139 IC50 = 18.7 nM T80975 CSL4Y5 155519270 IC50 = 180 nM T80975 CT6V3O 155519533 IC50 = 55.95 nM T80975 C9HEY1 155519702 IC50 = 14490 nM T80975 C3M6GZ 155519761 IC50 = 410 nM T80975 C4YJN9 155520341 IC50 = 1600 nM T80975 CU6Z5O 155520650 IC50 = 260 nM T80975 CDNO69 155520677 IC50 = 200 nM T80975 CTC34D 155520839 IC50 = 96.17 nM T80975 C80EJR 155521068 IC50 > 10000 nM T80975 CP5N6R 155521169 IC50 = 2500 nM T80975 CMWI40 155521404 IC50 = 86 nM T80975 CX18UM 155522654 IC50 = 92 nM T80975 CQS78C 155522775 IC50 = 4400 nM T80975 C3ST0D 155522792 IC50 = 86 nM T80975 CB50GK 155522849 IC50 = 86.84 nM T80975 CD2YM4 155523255 IC50 = 11.06 nM T80975 C70NHV 155523393 IC50 > 10000 nM T80975 CXFH76 155523422 IC50 = 3.56 nM T80975 COI15M 155523425 IC50 > 10000 nM T80975 CY6NE1 155523855 IC50 = 180 nM T80975 CBP7G1 155524105 IC50 = 300.42 nM T80975 CBSW02 155524123 IC50 = 34 nM T80975 CU1L0P 155524210 IC50 = 258.8 nM T80975 CG13QJ 155524262 IC50 = 450.7 nM T80975 CRP7Q6 155525519 IC50 = 270 nM T80975 CEV4D0 155526828 IC50 = 38.1 nM T80975 C72KLJ 155526893 IC50 = 3790 nM T80975 C8K3OI 155527167 IC50 = 260.64 nM T80975 CY5Z6A 155527325 IC50 = 443.8 nM T80975 CV9Y3X 155527350 IC50 = 7.63 nM T80975 C3GNP6 155527669 IC50 > 1000 nM T80975 C0KT3B 155527754 IC50 = 64.8 nM T80975 CQLF39 155527847 IC50 = 864.18 nM T80975 CEQ0F9 155528026 IC50 > 3000 nM T80975 CTD5R7 155528337 IC50 = 240 nM T80975 C9P2NQ 155528441 IC50 = 340 nM T80975 COZ8F9 155529176 IC50 = 97.3 nM T80975 CLEJ03 155529517 IC50 = 710 nM T80975 CZAQ19 155529778 IC50 = 190 nM T80975 C9EG5P 155529832 IC50 = 542.2 nM T80975 CLJ5T9 155529954 IC50 = 183.56 nM T80975 CL0V4U 155530858 IC50 = 220 nM T80975 CT9CL6 155531062 IC50 = 4120 nM T80975 CIGX26 155531103 IC50 = 302 nM T80975 CJOL74 155531230 IC50 = 97 nM T80975 CZN1T8 155531589 IC50 = 96 nM T80975 CWO98B 155531773 IC50 = 3.6 nM T80975 CA0BC3 155531915 IC50 = 490 nM T80975 CI0L2U 155532703 IC50 = 221 nM T80975 C5H8ZR 155532737 IC50 = 4160 nM T80975 CX7F6L 155532789 IC50 = 101 nM T80975 C6ZE4H 155533175 IC50 = 230.1 nM T80975 C7OX2W 155533223 IC50 = 1883.43 nM T80975 C67XEV 155533571 IC50 > 3000 nM T80975 C6Y3HD 155533711 IC50 = 340 nM T80975 C3NZO0 155533789 IC50 = 280 nM T80975 C62QJP 155533965 IC50 = 396 nM T80975 C2DJ0A 155534253 IC50 = 460 nM T80975 CXY94L 155534355 IC50 = 10.56 nM T80975 C9UAB3 155534683 IC50 = 1100 nM T80975 C37RFQ 155534994 IC50 = 450 nM T80975 C3UT5M 155535028 IC50 > 10000 nM T80975 CMH2J4 155535076 IC50 = 67.84 nM T80975 C8HCT3 155535088 IC50 = 1960 nM T80975 CD8TO7 155535214 IC50 = 5150 nM T80975 CBO91T 155535319 IC50 = 73.7 nM T80975 C8H1CZ 155536201 IC50 = 330 nM T80975 CAL3C6 155536359 IC50 = 0.52 nM T80975 CT7XR2 155536438 IC50 = 3630 nM T80975 CF0A9O 155536643 IC50 > 1000 nM T80975 C3LC9I 155536820 IC50 = 6309.57 nM T80975 CDB1J4 155537585 IC50 = 740 nM T80975 C8S2CP 155537605 IC50 = 420 nM T80975 CKOC12 155537703 IC50 = 3200 nM T80975 CB6AN2 155537880 IC50 = 2510 nM T80975 C6PK7Q 155538522 IC50 = 1830 nM T80975 C35COQ 155538985 IC50 = 5500 nM T80975 C9RI7P 155539052 IC50 = 288.9 nM T80975 C65RJX 155539169 IC50 = 160 nM T80975 CS49XO 155539531 IC50 = 2270 nM T80975 CFEZ25 155539618 IC50 = 67 nM T80975 CEN71T 155539953 IC50 = 4082.09 nM T80975 C0HC7V 155540067 IC50 = 940 nM T80975 CWT25X 155540411 IC50 = 650 nM T80975 C4ZX8G 155540423 IC50 = 488.7 nM T80975 CE46SL 155540854 IC50 = 10770 nM T80975 C5O4JM 155540856 IC50 = 10500 nM T80975 CA5I7X 155541030 IC50 > 10000 nM T80975 C5N2ST 155541216 IC50 > 3000 nM T80975 C97AUG 155541960 IC50 = 4380 nM T80975 C9P3ON 155542000 IC50 = 15.9 nM T80975 C5Q3TM 155542204 IC50 = 34 nM T80975 CP67JN 155542393 IC50 = 36.78 nM T80975 CL7N0Q 155542435 IC50 > 10000 nM T80975 CUL39W 155542605 IC50 = 115 nM T80975 C1VJH0 155543634 IC50 = 25180 nM T80975 CQ17XT 155543872 IC50 = 61.2 nM T80975 CP4KT1 155544904 IC50 = 75.86 nM T80975 CK0X3N 155545235 IC50 = 200 nM T80975 C2I6HY 155545590 IC50 = 20.2 nM T80975 C4M2JT 155545755 IC50 = 19.4 nM T80975 C7NRO6 155545934 IC50 = 14 nM T80975 CJN15V 155546412 IC50 = 244.76 nM T80975 CSI83K 155546458 IC50 = 2865.05 nM T80975 CJK8O9 155546662 IC50 = 132 nM T80975 CRW83F 155546918 IC50 = 5410 nM T80975 C7SF2C 155547229 IC50 = 95 nM T80975 C3VX6K 155547248 IC50 = 54 nM T80975 C9E2KH 155547486 IC50 = 462.38 nM T80975 CL8X7V 155547722 IC50 = 517.33 nM T80975 CM8E5L 155548006 IC50 = 2510 nM T80975 C0P9CG 155548234 IC50 = 120 nM T80975 C9KJ5X 155548587 IC50 = 40400 nM T80975 CUTY40 155548640 IC50 = 383.61 nM T80975 CM6D4S 155548753 IC50 = 212 nM T80975 CUS5A3 155549314 IC50 > 500000 nM T80975 CQF73Y 155549371 IC50 = 290 nM T80975 CZGJ90 155549636 IC50 > 500000 nM T80975 CW34RN 155549665 IC50 = 51.9 nM T80975 CW37ZQ 155549914 IC50 = 480 nM T80975 CY6RU2 155549975 IC50 = 407.47 nM T80975 C6URZ7 155550475 IC50 = 560 nM T80975 CH95WO 155550617 IC50 > 3000 nM T80975 C0IK8P 155550720 IC50 = 190 nM T80975 CB2Q4M 155550927 IC50 = 207.04 nM T80975 C10GJP 155551126 IC50 = 578.8 nM T80975 C49SQG 155551406 IC50 > 1000 nM T80975 CRS02E 155551888 IC50 = 104 nM T80975 CKAG94 155551896 IC50 = 96 nM T80975 CN3GD4 155552925 IC50 = 5 nM T80975 C2VNW3 155553566 IC50 > 1000 nM T80975 CP1B4Z 155553636 IC50 > 10000 nM T80975 CAC31S 155553712 IC50 = 103 nM T80975 CY9T5X 155554019 IC50 = 306000 nM T80975 C1BQ0L 155554054 IC50 = 2730 nM T80975 CR9H1E 155554156 IC50 = 3950 nM T80975 CYO3B0 155554258 IC50 = 30.1 nM T80975 C1D2XE 155554380 IC50 = 51.4 nM T80975 CGVU70 155554426 IC50 = 25640 nM T80975 CWS1U9 155554482 IC50 > 10000 nM T80975 CJL3D2 155555429 IC50 = 5010 nM T80975 CFWV90 155555441 IC50 = 81 nM T80975 C7PNW9 155555625 IC50 = 117 nM T80975 CYEO53 155555708 IC50 = 460 nM T80975 CUA73V 155555832 IC50 = 510 nM T80975 CWDR07 155555935 IC50 = 5970 nM T80975 CDKF14 155556917 IC50 = 36.16 nM T80975 C5Q6ZT 155556944 IC50 = 232.6 nM T80975 C3BPZ9 155557063 IC50 = 11.07 nM T80975 C2XQ6C 155557323 IC50 = 160 nM T80975 CTR18O 155557674 IC50 = 7940 nM T80975 CP60UD 155557689 IC50 = 120 nM T80975 CJWZ08 155557846 IC50 = 3740 nM T80975 CZD71I 155558249 IC50 = 1196.59 nM T80975 C92NTS 155558433 IC50 = 82000 nM T80975 CWD8X0 155558928 IC50 > 10000 nM T80975 C7TQ4A 155558974 IC50 = 187 nM T80975 CV7H5S 155559048 IC50 = 40000 nM T80975 CU38IX 155559179 IC50 = 950 nM T80975 CO0ER7 155560513 IC50 = 1730 nM T80975 CP6GZ9 155560763 IC50 > 500000 nM T80975 C3ISX8 155560929 IC50 = 170 nM T80975 C87OUZ 155561574 IC50 = 987.7 nM T80975 CQ3VN2 155561716 IC50 = 10450 nM T80975 C8L6PM 155561965 IC50 = 1240 nM T80975 CZ7E4R 155561977 IC50 = 386.4 nM T80975 CKG6T0 155562060 IC50 = 3520 nM T80975 CWV62X 155562083 IC50 = 16 nM T80975 C68EPN 155562201 IC50 = 100 nM T80975 CC5F3I 155562216 IC50 = 27 nM T80975 C40IYS 155562258 IC50 = 22910 nM T80975 C9Z4AX 155562699 IC50 = 1900 nM T80975 C46OBE 155562913 IC50 = 286 nM T80975 C81JZW 155563388 IC50 = 170 nM T80975 C3N4KQ 155563637 IC50 = 109 nM T80975 CE6IV8 155563850 IC50 = 58.9 nM T80975 CU7Z0H 155564272 IC50 = 1104.22 nM T80975 C9WH0L 155564290 IC50 = 734.9 nM T80975 CFG6Z5 155564309 IC50 = 1.33 nM T80975 CD2XG9 155564539 IC50 > 10000 nM T80975 C2C8VR 155564618 IC50 = 1380 nM T80975 CM23DI 155565660 IC50 = 460 nM T80975 CA3BV5 155565694 IC50 = 5480 nM T80975 CN8DY1 155566015 IC50 = 842.4 nM T80975 C5V8WF 155566059 IC50 = 520 nM T80975 CY42EB 155566265 IC50 > 10000 nM T80975 C6S5RB 155567797 IC50 = 131 nM T80975 CX8I9K 155567999 IC50 = 30.5 nM T80975 CEL6Z4 155568027 IC50 = 4220 nM T80975 C0E8CV 155568098 IC50 = 280 nM T80975 CGX46E 155568143 IC50 = 418.7 nM T80975 CK10HA 155568167 IC50 = 490 nM T80975 CJ8WF2 155568386 IC50 = 109 nM T80975 C1HKP3 155568631 IC50 = 147.9 nM T80975 CZ9GJ1 155568910 IC50 = 44.9 nM T80975 C1S8ZB 155568922 IC50 = 8100 nM T80975 CXH6P0 155569339 IC50 = 80 nM T80975 C94IJB 10367131 IC50 = 3 nM T80975 CBWO68 49800164 IC50 = 186 nM T80975 CI8LX0 57976125 IC50 = 3 nM T80975 D00ATA 5908088 IC50 = 140 nM T80975 D00ERW 44444843 Ki > 8876 nM T80975 D00GVV 5329155 IC50 = 70 nM T80975 D00HVA 11624601 Ki > 8200 nM T80975 D00MCJ 5329369 IC50 = 355 nM T80975 D00TBD 10461815 IC50 = 200 nM T80975 D00YWZ 18450753 IC50 = 4900 nM T80975 D01LEV 22394620 IC50 = 15400 nM T80975 D02AOT 44394105 IC50 = 18 nM T80975 D02BXJ 46864270 IC50 = 2.3 nM T80975 D02RWK 44400432 IC50 = 4 nM T80975 D03BQI 3794 IC50 = 2800 nM T80975 D03DYT 3035817 IC50 = 43 nM T80975 D03DZO 11715767 IC50 > 10000 nM T80975 D03EHM 24905142 IC50 = 12 nM T80975 D03HLH 44331231 IC50 = 9800 nM T80975 D03HQK 5329843 IC50 = 870 nM T80975 D03HTT 44409370 IC50 = 10000 nM T80975 D04FNY 25195216 IC50 = 70 nM T80975 D04NGS 5330790 IC50 = 130 nM T80975 D04RQU 44425819 IC50 = 1000 nM T80975 D04ZWF 53396311 IC50 > 2000 nM T80975 D05NEC 60182364 IC50 = 1520 nM T80975 D05NKG 16760286 IC50 = 1000 nM T80975 D06BVH 18516979 IC50 = 1000 nM T80975 D06HVH 54613583 IC50 = 7200 nM T80975 D06LJL 9916282 IC50 = 1000 nM T80975 D06QWO 14824655 IC50 > 10 ug.mL-1 T80975 D06WGX 9549184 IC50 > 50000 nM T80975 D07AIB 712152 IC50 = 2720 nM T80975 D07IHM 9823787 IC50 > 3378 nM T80975 D07OCA 5330812 IC50 = 32 nM T80975 D07OXC 11650194 Ki = 422 nM T80975 D07SRX 9797919 Ki = 15 nM T80975 D08GBT 71295845 IC50 = 67 nM T80975 D08JSJ 1416020 IC50 = 1800 nM T80975 D08RZB 11153014 IC50 > 10000 nM T80975 D09AKX 1416247 IC50 = 1600 nM T80975 D09EAE 10131254 IC50 = 100 nM T80975 D09HVH 135566652 IC50 > 10 nM T80975 D09HXU 16086113 IC50 = 4966 nM T80975 D09LEK 5329850 IC50 = 500 nM T80975 D09LKM 5329468 IC50 = 19 nM T80975 D09LPL 5329103 IC50 = 27 nM T80975 D09QBA 23378546 IC50 = 4175 nM T80975 D09TNR 9850161 IC50 = 69 nM T80975 D09TQP 12043829 IC50 = 1200 nM T80975 D09XIL 11396738 IC50 = 50 nM T80975 D0A1CM 5281855 IC50 = 790 nM T80975 D0A4XJ 5289418 IC50 = 20 nM T80975 D0A9ZP 42609931 IC50 = 48 nM T80975 D0A9ZQ 5329846 IC50 = 1410 nM T80975 D0BM4F 5329404 IC50 = 134 nM T80975 D0BS6R 9549183 IC50 > 50000 nM T80975 D0BU6T 354471 IC50 = 500 nM T80975 D0C2GE 67161540 IC50 = 4 nM T80975 D0C6KI 5329006 IC50 = 100 nM T80975 D0CM6T 11314340 Ki > 3700 nM T80975 D0D3QA 44409436 IC50 = 270 nM T80975 D0D3YL 5329849 IC50 = 870 nM T80975 D0D6MH 11617559 IC50 > 20000 nM T80975 D0D9PD 11656591 IC50 > 5000 nM T80975 D0E3HC 5329450 IC50 = 3 nM T80975 D0E9DI 44430881 IC50 = 1000 nM T80975 D0EE6A 6398883 IC50 = 23 nM T80975 D0EU1R 46215815 IC50 > 10000 nM T80975 D0F0AU 44405988 IC50 = 17000 nM T80975 D0F2MP 60182389 IC50 = 5330 nM T80975 D0G3SZ 6918469 IC50 = 5 ug.mL-1 T80975 D0H1OK 11562302 IC50 = 130 nM T80975 D0H2CM 135565635 IC50 = 1500 nM T80975 D0IR6U 5494425 IC50 = 1400 nM T80975 D0J3LR 11634725 Ki > 4000 nM T80975 D0J3OZ 21934605 IC50 = 990 nM T80975 D0K6YK 11676119 IC50 = 2440 nM T80975 D0KH5T 5687 IC50 = 50 nM T80975 D0L0HG 766949 IC50 > 10000 nM T80975 D0L3FK 5289419 IC50 = 130 nM T80975 D0L3JR 25212148 IC50 = 5 nM T80975 D0M4QA 56935577 IC50 = 2.3 nM T80975 D0M4SY 135440466 IC50 = 1400 nM T80975 D0M9OF 5329371 IC50 = 8 nM T80975 D0ME9B 46868971 IC50 = 710 nM T80975 D0OZ2S 11785878 IC50 = 5100 nM T80975 D0PP6Y 60182393 IC50 = 1.68 nM T80975 D0Q3KS 9957049 IC50 > 5000 nM T80975 D0Q3NG 11715520 Ki > 8200 nM T80975 D0Q4EQ 16742063 IC50 = 11 nM T80975 D0Q5UH 9858940 IC50 > 10000 nM T80975 D0R2WK 16038120 EC50 > 1000 nM T80975 D0RF7O 44577753 IC50 = 19700 nM T80975 D0S7IE 11658882 Ki > 8200 nM T80975 D0ST4P 5187941 IC50 = 190 nM T80975 D0U3ZP 5329338 IC50 = 113 nM T80975 D0UN9O 3385203 IC50 >= 10000 nM T80975 D0US9O 45275255 IC50 = 22 nM T80975 D0UX3T 5329361 IC50 = 126 nM T80975 D0V9DQ 5329847 IC50 = 500 nM T80975 D0X1RH 16051023 IC50 = 1200 nM T80975 D0X6KS 16125109 IC50 > 12500 nM T80975 D0Y0BK 11524144 IC50 = 220 nM T80975 D0Y1SR 11844351 IC50 = 640 nM T80975 D0Y9GK 16125106 IC50 = 4790 nM T80975 D0YN1E 5329454 IC50 = 224 nM T80975 D0Z7TM 22273644 IC50 = 25 nM T80975 D0Z8TR 5298698 IC50 = 78 nM T59929 C89JSI 65245 IC50 = 30000 nM T59929 CIQ76Y 79516 IC50 > 100000 nM T59929 C6XA8R 100608 IC50 > 100000 nM T59929 CUR6F9 308653 IC50 = 148000 nM T59929 C9B8EM 309829 IC50 = 125000 nM T59929 C7BV2W 309844 IC50 = 30000 nM T59929 CV2LG4 451931 Ki = 236 nM T59929 C58TWR 490681 Ki = 236 nM T59929 CS05ZD 595027 IC50 = 30000 nM T59929 C2N4XS 6323266 Ki = 1.3 nM T59929 CJW05D 9561607 IC50 = 77000 nM T59929 CL0I3U 9903778 Ki = 17 nM T59929 C4YRV1 9949975 IC50 = 15100 nM T59929 CA8Z9S 10072342 IC50 > 200000 nM T59929 C1JLU4 10087523 IC50 = 1.9 nM T59929 C4X0WP 10087524 IC50 = 19 nM T59929 CD14AM 10105760 IC50 = 49 nM T59929 CEM21G 10181606 Ki = 770 nM T59929 C18PTM 10314206 IC50 = 20 nM T59929 CRIX75 10358357 IC50 = 24400 nM T59929 CT7Y0M 10470961 Ki = 64300 nM T59929 CQY2T5 10955570 IC50 = 257700 nM T59929 CX9CI2 11000363 IC50 = 21 nM T59929 CP57LN 11022009 IC50 = 21700 nM T59929 CLJ3D4 11160569 IC50 = 92400 nM T59929 CEG0Q5 11219482 IC50 = 200000 nM T59929 COPW05 11334014 IC50 = 143000 nM T59929 CDH37T 11336042 IC50 = 181000 nM T59929 CR1E3O 11347856 IC50 = 41000 nM T59929 CNS29Y 11432530 IC50 = 26000 nM T59929 C12GZY 11459028 IC50 = 500000 nM T59929 CR75CM 11482820 IC50 = 26000 nM T59929 CU8HS2 11746845 IC50 = 560 nM T59929 CIM8G0 11746846 IC50 = 100 nM T59929 CL81HQ 11819216 IC50 = 6300 nM T59929 CB6JA0 11829946 Ki > 20000 nM T59929 C54QHP 12255109 IC50 = 48977.88 nM T59929 C1AXR0 13115629 IC50 > 100000 nM T59929 C3WU0B 13740570 Ki > 20000 nM T59929 C3WE6Y 15908412 IC50 = 350 nM T59929 CZ39XW 16082761 IC50 = 24000 nM T59929 C26PWX 16082762 IC50 = 13000 nM T59929 C43IJY 16082763 IC50 = 19000 nM T59929 CLGB92 16082764 IC50 > 20000 nM T59929 C3A6PH 16082765 IC50 > 100000 nM T59929 CAB0D5 16082766 IC50 >= 40000 nM T59929 CV3J2I 16082771 IC50 > 75000 nM T59929 CE6J3S 16082772 IC50 = 45000 nM T59929 C3DJ0F 16082775 IC50 = 49000 nM T59929 CJ76DK 16082778 IC50 = 137000 nM T59929 CW0R4Q 16082779 IC50 = 23000 nM T59929 C8C2OJ 16098970 Ki = 43500 nM T59929 C86KQA 16098971 Ki = 8030 nM T59929 CLT64W 16098972 Ki = 1050 nM T59929 C5D1RX 16098980 Ki > 500000 nM T59929 CB18VS 16098981 Ki = 33400 nM T59929 CUV95Q 23648514 Ki = 200 nM T59929 CZXH68 23648515 Ki = 420 nM T59929 CWC6V4 23648516 Ki = 3340 nM T59929 CG65LC 23648517 Ki = 490 nM T59929 CCGO91 23648519 Ki = 1270 nM T59929 CU7I4R 23648520 Ki = 3940 nM T59929 C90GWS 23648521 Ki = 710 nM T59929 C9RB7M 23648524 Ki = 1170 nM T59929 C4AX1K 23648525 Ki = 630 nM T59929 COV4H8 23648526 Ki = 410 nM T59929 CCD5E6 23648529 Ki > 20000 nM T59929 CZHW05 23648530 Ki > 20000 nM T59929 C0OSI2 23730934 Ki = 3010 nM T59929 C81QDB 44268116 Ki > 300000 nM T59929 CIPM63 44268149 Ki > 600000 nM T59929 CO4U7K 44418782 Ki = 236 nM T59929 CV3D1U 45102605 IC50 = 13090 nM T59929 C38TLG 45263333 IC50 = 2200 nM T59929 CS6TW1 45263336 IC50 = 7500 nM T59929 CN7CF1 45263337 IC50 = 5000 nM T59929 CU38NG 45263340 IC50 = 7500 nM T59929 C2ZVX3 45263342 IC50 = 7000 nM T59929 CYJ67D 45263346 IC50 = 7400 nM T59929 C9KW6N 45263350 IC50 = 7200 nM T59929 CF0W5C 45263375 IC50 = 6300 nM T59929 C0QG8M 45263376 IC50 = 4600 nM T59929 C4IYO3 45263380 IC50 = 12100 nM T59929 CA53FU 45263385 IC50 = 7000 nM T59929 C4GRJ8 45263386 IC50 = 8000 nM T59929 C1EP4I 45263388 IC50 = 7400 nM T59929 CFOA29 45265816 IC50 = 8200 nM T59929 CLN42U 45265826 IC50 = 4600 nM T59929 C3I0TQ 45265843 IC50 = 3600 nM T59929 C6J1TH 45265845 IC50 = 6000 nM T59929 CQJ16N 45265846 IC50 = 8000 nM T59929 C2MVJ7 45266043 IC50 = 3800 nM T59929 C40LUI 46231938 Ki = 236 nM T59929 C5RQ6E 46231939 Ki = 236 nM T59929 CG4ZR0 46232010 Ki = 236 nM T59929 C1BXN4 49795955 Ki = 76000 nM T59929 C9YE2F 49795956 Ki > 2400000 nM T59929 CQWI30 51003442 IC50 = 17000 nM T59929 CD10FY 53320656 IC50 = 23000 nM T59929 C5M4CG 58448315 IC50 = 39560 nM T59929 C2JSY1 71741142 IC50 = 55700 nM T59929 CKV18J 71814332 IC50 = 22060 nM T59929 CFN5O6 72374609 IC50 = 9920 nM T59929 C24VAE 72374610 IC50 = 8540 nM T59929 CA0C6Q 72374611 IC50 = 13710 nM T59929 C5LQS9 72374612 IC50 = 22430 nM T59929 C5LYM3 72374613 IC50 = 19800 nM T59929 CFPQ85 72374614 IC50 = 33950 nM T59929 C6OGB0 72374615 IC50 = 33780 nM T59929 CL0X9J 72374616 IC50 = 64330 nM T59929 CTK2U4 72374617 IC50 = 2950 nM T59929 C9AWB7 72374710 IC50 = 36370 nM T59929 CXYK40 72376097 IC50 = 43320 nM T59929 C7W6VD 72376098 IC50 = 22630 nM T59929 CN4B0L 72376099 IC50 = 22140 nM T59929 CJA83H 72376100 IC50 = 30290 nM T59929 C4B0RW 72376101 IC50 = 31780 nM T59929 CVB1T2 72376102 IC50 = 48240 nM T59929 CAIL36 72376103 IC50 = 34420 nM T59929 C59FYO 72376104 IC50 = 23180 nM T59929 CX08IT 72376105 IC50 = 48540 nM T59929 CXZ8Q1 72376179 IC50 = 36560 nM T59929 CF98TP 72376180 IC50 = 22680 nM T59929 CN7MI4 72376181 IC50 = 25980 nM T59929 CYM92W 72376182 IC50 = 32210 nM T59929 CNC7H9 72376183 IC50 = 31580 nM T59929 CWC2F4 72376184 IC50 = 21910 nM T59929 C5XG7H 72376185 IC50 = 33060 nM T59929 C4PMI2 72376186 IC50 = 10840 nM T59929 C20ISE 72376187 IC50 = 21900 nM T59929 C1GNL6 72711417 IC50 > 100000 nM T59929 C7Q2UV 72711418 IC50 > 100000 nM T59929 C82QHN 72711419 IC50 > 100000 nM T59929 CE9V2K 86288857 Ki = 1770 nM T59929 CR52QW 86288858 Ki = 1650 nM T59929 C3DN2A 86288859 IC50 = 6109.42 nM T59929 C48VCT 86288860 IC50 = 4456.56 nM T59929 CFM5Z1 86288887 IC50 = 4285.49 nM T59929 CC0EY9 90654810 IC50 = 51522.86 nM T59929 CR1N8W 90654811 IC50 = 36720 nM T59929 C5B7LH 90654812 IC50 = 27669.42 nM T59929 CFLG62 90654813 IC50 = 30320 nM T59929 C4C9NU 90654814 IC50 = 29920 nM T59929 CD1Z6N 90654815 IC50 = 7533.56 nM T59929 C08OXN 90654816 IC50 = 14780 nM T59929 CY3H0B 90654817 IC50 = 22646.44 nM T59929 CR7MT1 90654818 IC50 = 19980 nM T59929 CFYV47 90654819 IC50 = 12560.3 nM T59929 CVP54W 90654820 IC50 = 51404.37 nM T59929 CGZX37 90654821 IC50 = 37380 nM T59929 CY80ZW 134130216 IC50 = 225670 nM T59929 CLHE72 134131196 IC50 = 61000 nM T59929 C0FB2A 134131292 IC50 = 65450 nM T59929 C4NWA7 135423677 IC50 = 94800 nM T59929 C3U8HB 135497173 IC50 = 18000 nM T59929 C1Q2IJ 135526599 IC50 = 30000 nM T59929 CYV94M 135541547 IC50 = 4500 nM T59929 C3JMR2 135541548 IC50 = 96000 nM T59929 C98ZJR 135541549 IC50 > 200000 nM T59929 CHI9K0 136233532 IC50 > 100000 nM T59929 C6J3CB 136233533 IC50 > 100000 nM T59929 C2YKV7 145979597 IC50 = 3400 nM T59929 C0L8PG 145979636 IC50 = 33400 nM T59929 CNG08T 145979747 IC50 = 25100 nM T59929 CF7PC1 145980985 IC50 = 16500 nM T59929 C30WPY 145981728 IC50 = 41300 nM T59929 CI72DM 145982043 IC50 = 41200 nM T59929 CC6Q5N 145985840 IC50 = 53700 nM T59929 CP3H8K 145987135 IC50 = 1400 nM T59929 CQBV80 145987666 IC50 = 85600 nM T59929 CIA05X 145987924 IC50 = 120 nM T59929 CH32UF 145988275 IC50 = 39900 nM T59929 CZH46L 145988451 IC50 = 2700 nM T59929 C4TNE7 145989148 IC50 = 15600 nM T59929 CY4R3F 145989768 IC50 = 15900 nM T59929 CK0V1U 145990719 IC50 = 10700 nM T59929 C0D9OB 145991688 IC50 = 37300 nM T59929 CJ17HV 145992132 IC50 = 22500 nM T59929 C0QC8M 145992338 IC50 = 44100 nM T59929 CJQ6Z8 145992671 IC50 = 21400 nM T59929 C20YPQ 145992892 IC50 = 7200 nM T59929 CUIZ59 145993844 IC50 = 25200 nM T59929 CIL9M2 145994177 IC50 = 49300 nM T59929 CQ35FA 155511213 IC50 = 36000 nM T59929 CLW31F 155513597 IC50 = 8400 nM T59929 C3ND8X 155513827 IC50 = 39000 nM T59929 CDU7H2 155517383 IC50 = 24000 nM T59929 CTU67Z 155524559 IC50 = 120 nM T59929 CYID76 155530666 IC50 > 100000 nM T59929 CGS16W 155532857 IC50 = 1200 nM T59929 COTC67 155533914 IC50 = 1000 nM T59929 C5F6UV 155535389 IC50 = 40000 nM T59929 C0JEP4 155544311 IC50 = 28000 nM T59929 C4UAF0 155551820 IC50 = 34000 nM T59929 CH1TK6 155562020 IC50 > 100000 nM T59929 C6Z1EM 155565310 IC50 = 87000 nM T59929 CK1Y7C 155565631 IC50 = 5600 nM T59929 D00PMF 45263378 IC50 = 3800 nM T59929 D01DAQ 44632008 Ki = 17 nM T59929 D01IGW 23648518 Ki = 400 nM T59929 D03IMY 23648512 Ki = 1060 nM T59929 D03ITH 16082760 IC50 = 4400 nM T59929 D04KCX 739395 IC50 = 38240 nM T59929 D04OWX 16082776 IC50 = 2300 nM T59929 D05OUP 16082758 IC50 = 13000 nM T59929 D06BMN 16082759 IC50 = 11000 nM T59929 D09TBA 23648513 Ki = 4550 nM T59929 D0A6LX 308654 IC50 > 200000 nM T59929 D0C0HN 23648522 Ki = 280 nM T59929 D0CO5S 23648511 Ki = 1790 nM T59929 D0DX8A 11095381 Ki = 4020 nM T59929 D0E7SH 23648510 Ki = 3090 nM T59929 D0E9PL 23648527 Ki = 470 nM T59929 D0G1DS 45263377 IC50 = 4300 nM T59929 D0I7IF 23648528 Ki = 1210 nM T59929 D0RE9X 14956545 Ki = 1030 nM T59929 D0VW6H 45265835 IC50 = 8300 nM T59929 D0W6LJ 16082777 IC50 = 11000 nM T59929 D0X5RA 80578 IC50 = 35 nM T59929 D0Y5UF 45263353 IC50 = 7200 nM T11824 D05YBZ 7083 Ki = 69 nM T11824 D05TPI 72276 IC50 >= 200000 nM T11824 D07SDQ 969516 IC50 = 3500 nM T11824 D0U2BH 65064 IC50 = 1800 nM T11824 C2KJI7 3883 Ki = 2.5 nM T11824 C0VAW3 13735 IC50 = 69 nM T11824 CYX3S5 65043 IC50 = 69 nM T11824 C39BCE 68275 IC50 < 3000 nM T11824 CO41FC 964143 Ki = 789.8 nM T11824 CJ0O1B 1588443 IC50 = 380 nM T11824 CO1ZV8 2306524 Ki = 522.1 nM T11824 CY28LS 5293755 Ki = 617.6 nM T11824 C5ZS3K 5713403 Ki = 528.5 nM T11824 CZ9Q1O 5928757 Ki = 362.5 nM T11824 CQ3S8L 6450842 Ki = 261.5 nM T11824 CFXW58 11631766 Ki = 1410 nM T11824 C7EBU1 11776207 IC50 > 10000 nM T11824 CLV24A 14214498 IC50 = 1400 nM T11824 C62KEJ 14837578 IC50 = 710 nM T11824 CN0Y8F 15504852 IC50 = 13 nM T11824 CN9U3G 16049314 IC50 = 246 nM T11824 CWUS28 22361008 IC50 > 10000 nM T11824 CCL0P8 24858429 IC50 = 1635 nM T11824 CYDL23 24952085 IC50 = 440 nM T11824 C1RB4M 24966387 IC50 = 1200 nM T11824 C0BN8L 42643531 IC50 = 4 nM T11824 CD80XQ 54581735 IC50 = 80 nM T11824 C4FZ5A 56950118 Ki = 13 nM T11824 C90MUF 57176479 Ki = 599 nM T11824 C2K6JT 57379031 EC50 = 24 nM T11824 CTA24H 57578199 IC50 = 1700 nM T11824 CC8ZH7 58660303 IC50 > 10000 nM T11824 CU1D5F 58795397 Ki = 797.8 nM T11824 CQU9W0 66556402 Ki = 191.3 nM T11824 CJ4R7E 66571561 IC50 = 660 nM T11824 CAJ6B8 67973277 EC50 = 325 nM T11824 C2ZCF9 67973354 EC50 = 169 nM T11824 C9JMF7 68551830 IC50 = 910 nM T11824 CXS67Z 68552247 IC50 = 580 nM T11824 CWE58F 68553100 IC50 = 690 nM T11824 CH54DU 68553676 IC50 = 600 nM T11824 CY8HE3 68553756 IC50 = 420 nM T11824 C1LYJ4 68553873 IC50 > 10000 nM T11824 CAG5N8 68554590 IC50 = 2000 nM T11824 CSQ53N 68555084 IC50 = 520 nM T11824 CEI5O1 68555350 IC50 = 320 nM T11824 CNCS47 68556083 IC50 = 1400 nM T11824 CN2QL6 68556085 IC50 = 920 nM T11824 CR4VM9 70686684 Ki = 1428 nM T11824 CD1PU4 70688786 Ki = 17 nM T11824 C59PES 70694381 Ki = 0.48 nM T11824 CZ3QF7 70697093 Ki = 112 nM T11824 CW0ZX3 71452100 IC50 = 2 nM T11824 CUP70I 71453931 IC50 = 1251 nM T11824 C7EX1K 71457447 IC50 = 17 nM T11824 CM5E3R 71457448 IC50 = 2 nM T11824 C3GPE7 71457449 IC50 = 4707 nM T11824 C7XML1 71457851 IC50 = 5.1 nM T11824 C4AK0O 71459256 IC50 = 42 nM T11824 CQ0FG2 71459258 IC50 = 7469 nM T11824 CYN3M8 71461086 IC50 = 1591 nM T11824 CW1E7U 71462763 IC50 = 6 nM T11824 CM6R2W 71463212 IC50 = 1.41 nM T11824 CLVB69 73294880 IC50 = 13 nM T11824 CGZK85 73296378 IC50 = 2 nM T11824 C9L3VR 73296809 IC50 = 2 nM T11824 C2S9PZ 73296810 IC50 = 5 nM T11824 C4XR1C 73297137 IC50 = 1 nM T11824 CCPI94 73297139 IC50 = 3 nM T11824 CE9X5J 86713212 IC50 = 420 nM T11824 C45CME 89681657 IC50 > 10000 nM T11824 C3R4PD 89970609 IC50 = 330 nM T11824 C06FNJ 89970660 IC50 = 610 nM T11824 CE1IW4 89970765 IC50 = 700 nM T11824 CEF8J5 90040128 IC50 = 5 nM T11824 CD48HU 90277509 IC50 > 10000 nM T11824 CX28SL 90644922 IC50 = 2 nM T11824 CHD0Z7 90644923 IC50 = 79 nM T11824 CYPJ75 90644924 IC50 = 8 nM T11824 CTL20G 102196384 IC50 > 10000 nM T11824 C5PBW3 102398558 IC50 > 10000 nM T11824 C5W7PM 118713185 IC50 > 10000 nM T11824 CQ07AH 118713186 IC50 > 10000 nM T11824 C5OFH2 118713187 IC50 > 10000 nM T11824 C9ZGB4 118713188 IC50 > 10000 nM T11824 C7Z2GA 118713189 IC50 > 10000 nM T11824 C03URO 118713190 IC50 > 10000 nM T11824 CYK30H 118713191 IC50 > 10000 nM T11824 CK53ME 118713192 IC50 > 10000 nM T11824 C35IDH 118713193 IC50 < 290 nM T11824 CM7UC8 118713194 IC50 > 10000 nM T11824 C5C8LX 118713195 IC50 = 300 nM T11824 C1RH3Y 118713196 IC50 = 1600 nM T11824 CB03DR 122182244 Ki = 212.4 nM T11824 CI6WT0 122182245 Ki = 431.7 nM T11824 C3X5KJ 122182246 Ki = 364 nM T11824 CT5G1Q 122182247 Ki = 1116.2 nM T11824 CCT7H6 122182248 Ki = 858.8 nM T11824 CML3T5 122182249 Ki = 853.5 nM T11824 CMO1C3 122182250 Ki = 169 nM T11824 CIT52U 122182251 Ki = 53.7 nM T11824 C19GJH 122182252 Ki = 35.1 nM T11824 CUOB01 122182253 Ki = 48 nM T11824 CW2V5B 122182254 Ki = 682.4 nM T11824 C75OCP 122182255 Ki = 717.6 nM T11824 CVH2T0 122182256 Ki = 229.1 nM T11824 CKQF12 122182257 Ki = 374 nM T11824 C7AUF8 122182258 Ki = 239.7 nM T11824 C7BXY4 122182259 Ki = 90 nM T11824 CCEL74 122182260 Ki = 188 nM T11824 C32GEV 122182261 Ki = 263.2 nM T11824 CWIT38 122182262 Ki = 257 nM T11824 CMVS36 122182263 Ki = 204.3 nM T11824 CLW95X 122182264 Ki = 131.1 nM T11824 C4TNB1 122182265 Ki = 465.1 nM T11824 CQ4R0K 122182266 Ki = 38.3 nM T11824 C5C8FY 122182267 Ki = 1756.7 nM T11824 C7NV9G 122182268 Ki = 27.1 nM T11824 CU3NJ6 122182269 Ki = 208.7 nM T11824 CS84HC 122182270 Ki = 121.5 nM T11824 C8EYO3 122182271 Ki = 590.5 nM T11824 CFV32E 122182272 Ki = 72.4 nM T11824 C1LHQ2 122182273 Ki = 318.1 nM T11824 C24PHB 122182274 Ki = 228.6 nM T11824 C1U3FZ 122182275 Ki = 354.6 nM T11824 CX5NB4 122182276 Ki = 151.7 nM T11824 CAU9H6 122182277 Ki = 630.3 nM T11824 C2RB1F 122182278 Ki = 80.1 nM T11824 CTMV35 122182279 Ki = 455.7 nM T11824 CO54NG 134133007 IC50 = 230 nM T11824 C4G8CN 136259624 IC50 = 970 nM T11824 C0PX2K 145968691 IC50 = 12900 nM T11824 C4R3UA 145978145 IC50 = 27200 nM T11824 CYB0T8 155552280 Ki = 120 nM T11824 D05CCT 4139 EC50 = 130 nM T11824 D0O5FK 10171487 IC50 = 3255 nM T11824 D0T3PW 5281672 IC50 = 1200 nM T11824 D0Z7EL 5280647 IC50 < 3000 nM T92724 D04AIT 5280445 IC50 = 20000 nM T92724 D07EXH 359 IC50 > 200000 nM T92724 D07MGA 72281 IC50 = 8300 nM T92724 D0J9ZR 4477 IC50 = 40000 nM T92724 D0K8KX 5280343 IC50 = 8100 nM T92724 C5H9TY 14697 IC50 = 207000 nM T92724 C3I7VB 102678 IC50 = 24500 nM T92724 CL5Y4J 159516 Ki = 3100 nM T92724 CV0B7W 442027 IC50 = 49600 nM T92724 C1E2FR 442048 IC50 = 283500 nM T92724 CZ3MD8 647122 IC50 = 16100 nM T92724 C2C8QU 948801 Ki = 27500 nM T92724 CXA4P6 1265413 IC50 = 90720 nM T92724 CUD4A1 1328543 IC50 = 58350 nM T92724 C3ZP4U 2131972 Ki = 9110 nM T92724 CA1N3H 2131982 Ki = 9930 nM T92724 CKL8B2 2219105 IC50 = 29900 nM T92724 CN43XQ 2806068 IC50 = 160 nM T92724 C5J6MO 2849659 IC50 = 28800 nM T92724 CN3P7A 2911959 IC50 = 74500 nM T92724 CZDG23 2947583 IC50 = 186000 nM T92724 CBIP72 2986413 IC50 = 76700 nM T92724 CCU3P7 3635406 IC50 = 2200 nM T92724 CZF0R5 4004950 IC50 = 500 nM T92724 C3AN7C 4117477 IC50 = 1180 nM T92724 CS2WB7 4236803 IC50 = 29800 nM T92724 C0AW3N 4378077 IC50 = 13860 nM T92724 CO3Y0T 4614896 IC50 = 9910 nM T92724 CY68ZT 4788586 IC50 = 940 nM T92724 CTR4Q1 5320532 IC50 = 13300 nM T92724 CVG47I 5958938 IC50 = 10500 nM T92724 CD8ZT2 6026688 IC50 > 50000 nM T92724 C3LZX9 8027611 IC50 = 12660 nM T92724 CJ4C5K 9180583 IC50 = 10800 nM T92724 CYQ8Z4 9882716 IC50 > 50000 nM T92724 C8K2NO 10062715 IC50 = 800000 nM T92724 C49CMU 10411574 IC50 = 21700 nM T92724 C6GN2F 11642725 IC50 = 870000 nM T92724 CHYP53 12310492 IC50 = 233400 nM T92724 C65EOH 15949840 IC50 = 7500 nM T92724 C9V8EM 15956553 IC50 = 300000 nM T92724 C3WYR4 16061499 IC50 = 2000 nM T92724 CTO43V 16085283 Ki = 116000 nM T92724 CU35DQ 21582568 IC50 = 220800 nM T92724 CN45FL 23427055 IC50 = 164700 nM T92724 CK3AF8 25256829 IC50 = 5400 nM T92724 C2SZ7L 42624533 IC50 = 14000 nM T92724 CYP8V1 44404067 IC50 > 50000 nM T92724 CD20PF 44433696 IC50 = 80000 nM T92724 CI4P2V 44433697 IC50 = 10000 nM T92724 CW7B0J 44433698 IC50 = 15000 nM T92724 C8DWL3 44433699 IC50 = 200000 nM T92724 C0ZPE2 44517748 IC50 = 2700 nM T92724 C0OH2T 44584893 IC50 = 5400 nM T92724 C0NZ5E 44584944 IC50 = 7300 nM T92724 CT70DZ 44590821 IC50 = 22500 nM T92724 C0SW2K 45266425 IC50 = 2500 nM T92724 C5WBP2 45266482 IC50 = 3800 nM T92724 CA4K8F 45266488 IC50 = 6600 nM T92724 C3BHZ4 45268445 IC50 > 50000 nM T92724 CC05NI 45268452 IC50 = 15400 nM T92724 C6QD9E 45269292 IC50 > 50000 nM T92724 CY7RV4 45269761 Ki = 21000 nM T92724 CO80TH 45269762 Ki = 297000 nM T92724 CU34ZK 45269763 Ki = 584000 nM T92724 C9P3LZ 45269764 Ki = 478000 nM T92724 CXS19V 45269765 Ki = 45200 nM T92724 C3DY4T 45270971 IC50 > 50000 nM T92724 CR4WA8 45270979 IC50 = 20900 nM T92724 CM78GO 45271412 Ki = 462000 nM T92724 CC90BU 45271826 IC50 = 5200 nM T92724 C0B6KX 45271831 IC50 = 9300 nM T92724 CN85IQ 45271832 IC50 = 8100 nM T92724 C7IF2O 45272299 Ki = 363000 nM T92724 CZRV73 45272304 Ki = 34100 nM T92724 CGV14L 45272305 Ki = 112000 nM T92724 CVTL97 45272306 Ki = 2200 nM T92724 CAM89I 45273174 Ki = 135000 nM T92724 CZT67B 45273179 Ki = 614000 nM T92724 CHF4M5 45273180 Ki = 49300 nM T92724 CND1R3 45273184 Ki = 159000 nM T92724 C0V5WT 45273625 IC50 > 50000 nM T92724 C6OE7V 46784066 IC50 = 28300 nM T92724 C6LH5I 46881919 Ki = 800 nM T92724 CI2FO1 49870840 IC50 = 5500 nM T92724 CF2D0I 49870841 IC50 = 8400 nM T92724 CM52SZ 49870842 IC50 = 6800 nM T92724 C8Q2CZ 50885062 IC50 > 50000 nM T92724 CJ6KV7 52941131 IC50 = 13900 nM T92724 C8M2QD 52943127 IC50 = 24300 nM T92724 CQ84MD 52945913 IC50 = 12000 nM T92724 CJ1LG2 52945915 IC50 = 42000 nM T92724 CZ35DX 52945977 IC50 = 128900 nM T92724 CAB1Y3 52946772 IC50 = 163200 nM T92724 CO4R1B 52947200 IC50 = 18000 nM T92724 CC4X1O 52948928 IC50 = 137700 nM T92724 CMG4U7 52949213 IC50 = 10800 nM T92724 C0X5BL 58589722 IC50 = 76740 nM T92724 CY3CL6 71544384 IC50 = 610 nM T92724 CV3P2U 71544385 IC50 = 230 nM T92724 CJS60O 71571220 IC50 = 49000 nM T92724 C1AY0M 71571221 IC50 = 49000 nM T92724 CY21XB 71571222 IC50 = 4600 nM T92724 C1DX9H 71571223 IC50 = 39000 nM T92724 CKE2C3 73056463 IC50 > 100000 nM T92724 C9S8ZH 73056464 IC50 > 100000 nM T92724 CK9OI0 73056465 IC50 = 31710 nM T92724 C4D8LK 73056466 IC50 = 32080 nM T92724 CRY86G 73056467 IC50 = 34910 nM T92724 C3VS4F 73056760 IC50 = 10070 nM T92724 CYH1F4 73056761 IC50 = 51330 nM T92724 C2CRZ8 73056762 IC50 = 2250 nM T92724 CD4YR3 73056763 IC50 = 11830 nM T92724 C3P2OZ 73056764 IC50 = 67200 nM T92724 C1H8PX 73056765 IC50 = 82910 nM T92724 C8JO7B 73056766 IC50 = 13860 nM T92724 CCYE63 73057087 IC50 = 5520 nM T92724 C54JWM 73057088 IC50 = 39870 nM T92724 C8RBU6 73057089 IC50 = 1040 nM T92724 CEBH65 73057090 IC50 = 1690 nM T92724 C8M2DX 73057091 IC50 = 17820 nM T92724 CQ42AZ 73057092 IC50 = 2820 nM T92724 CPLJ64 73057388 IC50 = 4700 nM T92724 CIN5V0 76320984 IC50 = 4300 nM T92724 C05AYV 102341658 IC50 = 16400 nM T92724 C8S3CR 102341659 IC50 = 37500 nM T92724 C2G9CP 127043455 IC50 = 20200 nM T92724 CVZ4I3 127043641 IC50 = 6000 nM T92724 C7BST4 127043642 IC50 = 5800 nM T92724 CGO01F 127043643 IC50 > 50000 nM T92724 C2TU5A 127043644 IC50 = 6400 nM T92724 C0Y9IT 127043645 IC50 = 41200 nM T92724 CF3B1Z 127045220 IC50 = 11700 nM T92724 CIXJ94 127045221 IC50 = 8600 nM T92724 CQ1CT5 127045222 IC50 = 18700 nM T92724 CKRX04 127045227 IC50 = 30700 nM T92724 CDZ2E1 127045228 IC50 > 50000 nM T92724 CG3E9B 127045229 IC50 = 6700 nM T92724 CG6VR3 127045386 IC50 = 15700 nM T92724 CK9JE3 127045387 IC50 > 50000 nM T92724 CY1E4Z 127045392 IC50 > 50000 nM T92724 CK5PA4 127045393 IC50 = 44700 nM T92724 C34TWD 127045394 IC50 > 50000 nM T92724 C97MQC 127048409 IC50 = 20000 nM T92724 C41VRM 127048410 IC50 = 7500 nM T92724 CZ0B1R 127052510 IC50 = 10000 nM T92724 CRW05E 127052511 IC50 > 50000 nM T92724 CC3TX0 127052512 Ki = 72000 nM T92724 CIQ1U9 127052513 Ki = 41000 nM T92724 CI13JZ 135452883 IC50 = 10000 nM T92724 CG1KW5 135470831 IC50 = 77090 nM T92724 CH4Q6A 145964401 IC50 = 5500 nM T92724 CHU61S 145964420 IC50 = 42100 nM T92724 C6YCA8 145964710 IC50 = 28800 nM T92724 CV6F7L 145966788 IC50 = 2100 nM T92724 CBWX17 145967285 IC50 = 4300 nM T92724 COR9X3 145972736 IC50 = 3900 nM T92724 CQ0M2X 145972809 IC50 = 4100 nM T92724 CF95RZ 145972878 IC50 = 3200 nM T92724 CXI0D1 145975081 IC50 = 6300 nM T92724 CG84ZR 145975487 IC50 = 5100 nM T92724 C91FOT 145976006 IC50 = 5200 nM T92724 C3F4UH 145978039 IC50 = 8800 nM T92724 CL7FB0 2919450 IC50 = 62790 nM T92724 D00RIX 5280443 IC50 = 280800 nM T92724 D01XMM 4117383 IC50 = 4450 nM T92724 D08MZY 145937 Ki = 8200 nM T92724 D08UYP 3008868 Ki = 2400 nM T92724 D09BUG 10207 IC50 = 132000 nM T92724 D0L7AT 10480940 Ki = 19300 nM T92724 D0S0BN 130976 Ki = 10600 nM T92724 D0SY2M 5281708 IC50 = 105000 nM T92724 D0UQ6U 10569 IC50 = 189100 nM T92724 D0WA9S 10429214 IC50 = 146500 nM T88285 D02HFD 124886 Ki = 954992.59 nM T88285 D03XYW 3342 Ki = 383000 nM T88285 D04AIT 5280445 IC50 = 7700 nM T88285 D09BHB 5509 Ki = 87800 nM T88285 D0K8KX 5280343 IC50 = 3200 nM T88285 D0R1RS 3715 Ki = 18100 nM T88285 D0W9WF 3825 Ki = 414000 nM T88285 D0Z5IU 1548887 Ki = 77900 nM T88285 D07SDQ 969516 Ki = 5 nM T88285 D0ZN1R 68245 IC50 = 1900 nM T88285 D06EDT 1613 Ki = 1.2 nM T88285 D0SU1G 5733 Ki = 107000 nM T88285 C8R4QL 1981 Ki = 12900 nM T88285 CI9TK0 3884 Ki = 37153.52 nM T88285 C2HNF8 8369 Ki = 223872.11 nM T88285 CV2U6G 36591 IC50 > 200000 nM T88285 CL1Y4H 68247 IC50 = 11700 nM T88285 CB8M5R 95990 Ki = 91000 nM T88285 CN76GF 115260 Ki = 4168693.83 nM T88285 C2OM1U 151506 IC50 = 18500 nM T88285 CFO0Z8 161167 IC50 = 8500 nM T88285 CT09IW 240414 Ki = 383000 nM T88285 CYFI62 303544 Ki = 12900000 nM T88285 CJSM92 303545 Ki = 5500000 nM T88285 CXO7Q3 312235 Ki = 6300000 nM T88285 CRM1C5 312236 Ki = 8200000 nM T88285 C1WAC5 315100 Ki = 34700000 nM T88285 CWVQ13 315101 Ki = 38600000 nM T88285 C3EF4W 315102 Ki = 29600000 nM T88285 CQ73XA 374648 Ki = 160 nM T88285 CSM6F4 375165 Ki = 14 nM T88285 CH54TS 392749 Ki = 46 nM T88285 C7HME8 439246 Ki = 17378.01 nM T88285 C8KHF3 706495 IC50 > 200000 nM T88285 C2X5CF 721421 IC50 = 93200 nM T88285 CL7HM5 736681 Ki = 385000 nM T88285 CX43LR 923602 Ki = 1394000 nM T88285 CA76JS 958751 Ki = 1907000 nM T88285 C96RSV 1311294 IC50 = 3600 nM T88285 CK17WZ 1550161 Ki = 65000 nM T88285 C3XSU5 2306193 IC50 = 54600 nM T88285 C1XRI2 2848041 IC50 = 14500 nM T88285 CJO73U 3830428 IC50 = 5700 nM T88285 CCO1X8 4202587 Ki = 426000 nM T88285 CJ8LZ1 4215345 IC50 = 7000 nM T88285 CZ4NJ7 4349112 IC50 > 20000 nM T88285 CZX61N 4370641 IC50 = 1190 nM T88285 C0P3NT 4409074 Ki = 27000 nM T88285 CE3MA8 5006190 IC50 = 4200 nM T88285 CMAH08 5315472 Ki = 18000 nM T88285 C1TA0H 5326751 Ki = 10 nM T88285 C7FK3U 5380187 Ki = 11220.18 nM T88285 CP0WX3 5388618 Ki = 159000 nM T88285 CKD26W 7062472 IC50 = 2000 nM T88285 CE56QK 8823663 IC50 = 7500 nM T88285 CDW12O 8823695 IC50 = 7600 nM T88285 C42LEW 8823700 IC50 = 7300 nM T88285 CO3PB8 8823701 IC50 = 6600 nM T88285 CO3QD4 8823727 IC50 = 6600 nM T88285 CVKN50 10073735 Ki = 15500 nM T88285 CTQA53 10433984 Ki = 15848.93 nM T88285 C78UMQ 10737607 Ki = 183000 nM T88285 CNZ1Q2 11716566 Ki = 18000 nM T88285 CF23IW 11779786 Ki = 230 nM T88285 CSPD18 14368897 Ki = 478630.09 nM T88285 CH2MY8 16153598 Ki = 0.96 nM T88285 CV96DU 16759528 IC50 > 20000 nM T88285 CM69DG 16759534 IC50 > 20000 nM T88285 C2F4JN 22670868 IC50 > 20000 nM T88285 C1F5JU 22974334 IC50 = 1300 nM T88285 C5Z6QA 25038243 IC50 = 11200 nM T88285 C6QRB2 28046592 IC50 > 20000 nM T88285 CN4FS2 44195235 Ki = 3600 nM T88285 C9KM8I 44223450 IC50 = 53.9 nM T88285 C6F7KE 44279136 Ki = 28183.83 nM T88285 C1GD7N 44279138 Ki = 7585.78 nM T88285 CSXY18 44279161 Ki = 194984.46 nM T88285 CE80ON 44279232 Ki = 48977.88 nM T88285 C9RVQ5 44279252 Ki = 32359.37 nM T88285 CN4IA9 44279267 Ki = 27542.29 nM T88285 CBY90R 44279301 Ki = 93325.43 nM T88285 CZNM01 44279304 Ki = 39810.72 nM T88285 CE27OW 44279305 Ki = 8912.51 nM T88285 CPXK95 44279347 Ki = 7943.28 nM T88285 CD5BM1 44279352 Ki = 38904.51 nM T88285 CC9X1G 44279353 Ki = 100000 nM T88285 CCE89N 44279365 Ki = 30199.52 nM T88285 C4GXI2 44279387 Ki = 9772.37 nM T88285 C0KM3B 44279388 Ki = 7762.47 nM T88285 CICZ64 44279427 Ki = 10000 nM T88285 CT52PC 44279440 Ki = 10471.29 nM T88285 CLD31O 44279578 Ki = 74131.02 nM T88285 CA35NB 44279579 Ki = 11481.54 nM T88285 CC0JZ1 44279597 Ki = 67608.3 nM T88285 CRA49J 44279598 Ki = 20892.96 nM T88285 CP8G2C 44279622 Ki = 37153.52 nM T88285 CPFT52 44279638 Ki = 51286.14 nM T88285 CULX04 44279640 Ki = 194984.46 nM T88285 C83IXT 44279660 Ki = 436515.83 nM T88285 COR3M8 44279707 Ki = 93325.43 nM T88285 CL8S2J 44279747 Ki = 269153.48 nM T88285 C9VJD1 44279748 Ki = 24547.09 nM T88285 CKIN84 44308536 Ki = 1980000 nM T88285 C75LKI 44308565 Ki = 1700 nM T88285 COI65F 44308724 Ki = 2230000 nM T88285 CTIV58 44308763 Ki = 5670000 nM T88285 C05ZNY 45147309 IC50 > 200000 nM T88285 C49JCG 46175389 IC50 = 3900 nM T88285 C5UHD4 46887816 IC50 = 43000 nM T88285 CTX0W3 47177602 IC50 > 20000 nM T88285 C4U0VN 49850572 Ki = 3200 nM T88285 CQ14FV 49852108 Ki = 4600 nM T88285 CKC75X 49852110 Ki = 2600 nM T88285 CLFX79 51238103 IC50 > 20000 nM T88285 CE2ZW3 52106067 IC50 > 200000 nM T88285 CG3Z7N 53318274 Ki = 3600 nM T88285 CG4C3T 53323608 Ki = 39000 nM T88285 CN03IM 57407714 IC50 = 90000 nM T88285 C39TCB 57917839 IC50 > 200000 nM T88285 CGI5T1 59191097 IC50 = 6100 nM T88285 CJT1W3 59191107 IC50 > 20000 nM T88285 CP47FA 68183385 IC50 = 6900 nM T88285 CEU2X1 70679296 Ki = 11 nM T88285 CGJ63L 71450394 IC50 = 250 nM T88285 C0KY4C 71452217 IC50 = 8130 nM T88285 C6JGN3 71454021 IC50 = 300 nM T88285 CLJ9U3 71454022 IC50 = 300 nM T88285 CU28XL 71454023 IC50 = 40 nM T88285 CAR1B0 71455760 IC50 = 510 nM T88285 CB7AK3 71455761 IC50 > 10000 nM T88285 C2D0WG 71457549 IC50 > 10000 nM T88285 C5FAS0 71461177 IC50 = 260 nM T88285 CJX8I2 71461178 IC50 = 1520 nM T88285 C8I7ES 71461179 IC50 = 8280 nM T88285 C3FTZ8 71461180 IC50 = 8400 nM T88285 C42ONV 71461181 IC50 = 14 nM T88285 C8NXJ0 71462921 IC50 = 280 nM T88285 C4DY3Q 71462922 IC50 = 480 nM T88285 CQR5P1 84358281 IC50 = 8700 nM T88285 CQ51YR 84358282 IC50 = 4600 nM T88285 C78WCJ 87057567 Ki = 1 nM T88285 CI8CW3 90667458 IC50 = 26.4 nM T88285 CZB03X 90667459 IC50 = 51.3 nM T88285 C8FYE1 90667460 IC50 = 45.8 nM T88285 C83MWI 118873474 IC50 = 11500 nM T88285 CQUR74 118873479 IC50 > 20000 nM T88285 CL2DM7 122194037 Ki = 1 nM T88285 CD1K9W 122194038 Ki = 0.3 nM T88285 CFB9K3 122194039 Ki = 330 nM T88285 CO5H2A 122194040 Ki = 130 nM T88285 C17FAK 122194041 Ki = 46 nM T88285 CSUE76 153156039 IC50 > 100000 nM T88285 CVKH48 155510386 IC50 > 20000 nM T88285 CJAX10 155514797 IC50 = 3900 nM T88285 CIWM69 155516481 IC50 > 100000 nM T88285 C7CW4J 155520327 IC50 = 11200 nM T88285 CWC86Y 155521422 Ki = 7 nM T88285 C8K7IN 155524148 IC50 = 1320 nM T88285 C80AQX 155525914 IC50 = 540 nM T88285 CC4VU0 155530785 IC50 = 6200 nM T88285 C0G9IU 155531520 IC50 = 720 nM T88285 CO01YR 155532738 IC50 = 1210 nM T88285 C40QRT 155539326 IC50 = 790 nM T88285 CX41SB 155540175 IC50 = 460 nM T88285 C4N0RF 155546581 IC50 = 790 nM T88285 CYR8P1 155549907 IC50 = 500 nM T88285 C4EX8A 155551658 IC50 = 480 nM T88285 CJ8YQ2 155553290 IC50 = 5500 nM T88285 COUK87 155555757 IC50 = 13900 nM T88285 CFO87T 155557815 IC50 = 370 nM T88285 C4UI1Z 155557859 Ki = 19 nM T88285 C6MNI0 155560544 IC50 = 11900 nM T88285 C8JO5C 155562765 IC50 = 590 nM T88285 CM36XL 155563395 IC50 = 640 nM T88285 C1Q3RV 155564267 IC50 = 1190 nM T88285 C6ELG9 155565369 IC50 = 1040 nM T88285 CL5OU1 155569599 IC50 = 15400 nM T88285 CS95RC 390758 Ki = 1900 nM T88285 C9JQY1 390759 IC50 = 140500 nM T88285 C3NS7M 390760 Ki = 92900 nM T88285 C2K7RF 390761 IC50 = 1624600 nM T88285 CTL75N 44308719 Ki = 680000 nM T88285 C6N9WG 44308721 Ki = 3160000 nM T88285 D00XKH 10598311 Ki = 180 nM T88285 D00YEV 5281605 IC50 = 11000 nM T88285 D01UKL 10367177 Ki = 18 nM T88285 D01UYI 5281607 Ki = 83176.38 nM T88285 D03OXL 10740201 Ki = 800 nM T88285 D0E3VR 10574926 Ki = 170 nM T88285 D0FX3J 126845 Ki = 1700 nM T88285 D0G3TK 5280863 IC50 = 20600 nM T88285 D0I2AG 448107 Ki = 14 nM T88285 D0I6JQ 10322772 Ki = 46 nM T88285 D0I8PQ 10810621 Ki = 1180 nM T88285 D0MF5Y 5281614 Ki = 13182.57 nM T88285 D0NJ4H 5281670 Ki = 30199.52 nM T88285 D0O0VZ 667639 IC50 = 760 nM T88285 D0O3DI 67249 IC50 = 16400 nM T88285 D0R3IN 97537 Ki = 80 nM T88285 D0T3PW 5281672 IC50 = 560 nM T88285 D0X8OL 830459 IC50 = 4900 nM T88285 D0YI5C 10072462 Ki = 16 nM T88285 D0Z9WS 10411076 Ki = 14 nM T51191 D00SQN 12136798 IC50 = 110 nM T51191 D01QIN 60823 IC50 = 22547 nM T51191 D06WTZ 53232 IC50 = 25933 nM T51191 D09DHY 6167 IC50 > 20 ug.mL-1 T51191 D0E3SH 6918837 Ki = 0.65 nM T51191 D0E7PQ 5311 Ki = 1.6 nM T51191 D0L7LC 5352062 Ki = 0.038 nM T51191 D0Y3KG 3121 IC50 = 62000 nM T51191 D00FHR 9865515 Ki = 32.4 nM T51191 D01WKZ 53340426 IC50 = 318 nM T51191 D05KED 53340666 IC50 = 48 nM T51191 D06TKI 49857317 IC50 = 4 nM T51191 D07FPY 6918877 Ki = 36 nM T51191 D09XIZ 11538455 Ki = 0.06 nM T51191 D0B3FV 6445533 Ki = 1.4 nM T51191 D0B7CH 4775 IC50 = 65000 nM T51191 D0E6UZ 54575456 IC50 = 1.6 nM T51191 D0GE5B 56654642 IC50 = 1280 nM T51191 D0GH3Q 9804992 Ki = 3 nM T51191 D0L2UQ 49855250 Ki = 16 nM T51191 D0M8FD 4261 Ki = 65 nM T51191 D0V0SL 11749858 Ki = 19 nM T51191 D0XT6W 6918638 Ki = 0.85 nM T51191 D0Z4RC 24756910 IC50 = 12.6 nM T51191 D0J8OC 5186 Ki = 2.2 nM T51191 D00HXJ 118884610 Ki = 774 nM T51191 D0CH8Q 56965342 IC50 = 30 nM T51191 D0L1NO 72722126 IC50 > 50000 nM T51191 D0N2DK 72710871 IC50 = 8 nM T51191 D0QX3G 71532921 IC50 = 4400 nM T51191 D0YN2T 86302836 IC50 > 50000 nM T51191 D0ZG5X 71811260 IC50 = 3610 nM T51191 D0N3SH 4996 Ki = 36000 nM T51191 D0W9NH 2746 IC50 = 147 nM T51191 CBIR94 10313 IC50 = 7910 nM T51191 C1N2KZ 88129 IC50 = 680000 nM T51191 CW70DI 211808 IC50 > 100000 nM T51191 CF60JA 220184 IC50 > 33330 nM T51191 CE45SU 247630 IC50 > 1000 nM T51191 CH1JD3 419176 IC50 = 9000 nM T51191 C0Y4WC 614947 Ki = 0.42 nM T51191 CU3HS2 1108280 IC50 > 100000 nM T51191 C96GFC 1798422 IC50 = 100500 nM T51191 C94IXC 2173124 IC50 = 8750 nM T51191 C58NGX 2175719 IC50 = 6450 nM T51191 CJCY71 2295078 IC50 = 3020 nM T51191 CG41FO 2423676 IC50 = 5350 nM T51191 CEO31B 2423687 IC50 = 5860 nM T51191 CK8I3T 3432579 IC50 > 33330 nM T51191 CZA83Y 4118131 IC50 = 2720 nM T51191 CV9JS5 4288771 IC50 > 33000 nM T51191 CN4M6D 5281220 IC50 = 38900 nM T51191 CSIJ53 5793932 IC50 = 5100 nM T51191 C2NA1H 5842785 IC50 > 5000 nM T51191 C18ENP 6918846 Ki = 39 nM T51191 C1RD7E 6918878 Ki = 1.5 nM T51191 CE9LP2 9543539 IC50 = 1590 nM T51191 CJ07ZA 9800555 IC50 = 160 nM T51191 CC0EU7 9828788 IC50 = 3.9 nM T51191 CH2LR4 9835152 IC50 = 381 nM T51191 CLYJ85 9848223 IC50 = 270 nM T51191 CSW4Y1 9891541 IC50 = 200 nM T51191 C81EYJ 9923508 IC50 = 3 nM T51191 CQG4V8 9924543 IC50 = 0.8 nM T51191 COLN58 9965621 IC50 = 607 nM T51191 CQDG65 10110195 IC50 = 200 nM T51191 CWA9R2 10135838 IC50 = 441 nM T51191 CL4C9H 10154438 Ki = 0.1 nM T51191 C7RC1E 10309899 IC50 = 9 nM T51191 C9OU5F 10464879 Ki = 0.13 nM T51191 CDY91S 10584105 Ki = 0.26 nM T51191 CSMT47 10728039 Ki = 0.81 nM T51191 CK8UV7 11019840 Ki = 0.06 nM T51191 C5P3EI 11167060 IC50 = 80 nM T51191 C8G5WP 11210533 IC50 = 9100 nM T51191 CYJ60V 11244651 IC50 = 16400 nM T51191 CI7W3O 11267278 IC50 = 6460 nM T51191 CM6ZW2 11279156 IC50 = 4640 nM T51191 CY34EQ 11393847 IC50 = 200 nM T51191 CB3N5M 11514394 IC50 = 321 nM T51191 CRZ7H2 11556677 IC50 = 18 nM T51191 C2F9NT 11558827 IC50 = 647 nM T51191 C9UN7F 11637884 IC50 = 14500 nM T51191 C24SBP 11657529 IC50 = 160 nM T51191 CQ32FV 11664499 IC50 = 4 nM T51191 CG9OC4 11682502 IC50 = 17.9 nM T51191 CYB26W 11688197 IC50 > 1000 nM T51191 CJ2UA0 11690271 IC50 = 3360 nM T51191 CC3GQ0 11700059 IC50 = 59 nM T51191 CU0M1E 11947684 IC50 = 3.9 nM T51191 C0QCW4 11988293 IC50 = 2300 nM T51191 C9G1BN 11993595 IC50 = 3900 nM T51191 CH5JS7 11993694 IC50 = 440 nM T51191 CJ94OC 12542182 Ki > 2500 nM T51191 C06UTF 13507024 IC50 = 16 nM T51191 C4XJ8M 13889849 Ki = 470 nM T51191 C1KR4L 14113324 IC50 > 50000 nM T51191 C15MQN 14113325 IC50 > 50000 nM T51191 C2D1KP 15983982 Ki = 21 nM T51191 C7DK5L 15984110 IC50 = 500 nM T51191 CHB82E 15986417 IC50 = 2640 nM T51191 C52EVH 15986418 IC50 = 590 nM T51191 C0GED2 15986506 IC50 = 220 nM T51191 CEL7P9 15986507 IC50 = 460 nM T51191 CS1QO9 15986509 IC50 = 1160 nM T51191 C5T1WF 16006672 IC50 = 313 nM T51191 CQGC05 16036765 IC50 = 170 nM T51191 CM3T2E 16049824 IC50 = 29 nM T51191 C30UFT 16066811 IC50 = 272 nM T51191 CFK8J5 16068056 Ki = 26 nM T51191 CMQP70 16068495 Ki = 33 nM T51191 CT84XO 16068594 Ki = 18 nM T51191 CF3ZG5 16068595 Ki = 18 nM T51191 CL60CA 16068912 Ki = 14 nM T51191 C9ZQB3 16095102 Ki > 5000 nM T51191 C80XYC 16095113 Ki > 5000 nM T51191 C6BGM2 16659535 IC50 = 460 nM T51191 CQI9N3 16659537 IC50 = 330 nM T51191 C5YFV9 16661453 IC50 = 1480 nM T51191 C8S5OX 16661455 IC50 = 560 nM T51191 CH67WF 16661458 IC50 = 460 nM T51191 CZ72YC 16661613 IC50 = 260 nM T51191 C8DZ1T 16661615 IC50 = 1480 nM T51191 CQV40I 16661617 IC50 = 1440 nM T51191 C5CIB4 16663079 IC50 = 640 nM T51191 CUG50I 16733294 IC50 = 156 nM T51191 CWO7V0 16733295 IC50 = 2580 nM T51191 C4W0PG 16733410 IC50 = 167 nM T51191 C0MO3Z 16733411 IC50 = 113 nM T51191 C3QL4X 16733412 IC50 > 30000 nM T51191 CV54SY 16733414 IC50 = 1250 nM T51191 C1VCX2 16733415 IC50 = 492 nM T51191 CXN07K 16733416 IC50 > 30000 nM T51191 CP9AR8 16733417 IC50 = 205 nM T51191 CUE62T 16733590 IC50 > 30000 nM T51191 CB4IN2 16773791 IC50 = 2200 nM T51191 CQHD27 20459443 IC50 = 1050 nM T51191 CE2W3M 21630365 IC50 = 4800 nM T51191 CS5R0U 22836624 Ki = 12500 nM T51191 CD16PI 23521584 IC50 = 330 nM T51191 CB8A5Q 23648260 IC50 = 6 nM T51191 C1JZ6D 23648261 IC50 = 100 nM T51191 CQJS61 23648262 IC50 = 60 nM T51191 C35ILE 23648263 IC50 = 70 nM T51191 C82BVC 23648264 IC50 > 10000 nM T51191 CT6NY2 23648265 IC50 > 10000 nM T51191 CZV0Q2 23648266 IC50 = 60 nM T51191 C36NKL 23648268 IC50 = 200 nM T51191 C5YBX0 23760408 IC50 = 5000 nM T51191 CM73VT 23818230 IC50 = 2.1 nM T51191 CVAB64 23846833 IC50 = 3600 nM T51191 C8RC9P 24744325 IC50 = 45 nM T51191 CVB7J3 24746434 IC50 = 44 nM T51191 C28AWJ 24746436 IC50 = 71 nM T51191 C17GDO 24779722 IC50 >= 50 nM T51191 CA7O1E 24779723 IC50 >= 50 nM T51191 CIO7Q6 24853792 IC50 = 880 nM T51191 CBN0J5 24853793 IC50 = 110 nM T51191 CLT5J2 24881257 IC50 = 679 nM T51191 C5GCM1 24881328 IC50 = 294 nM T51191 C8QVB1 24881329 IC50 = 143 nM T51191 CU0AM3 24881330 IC50 = 43 nM T51191 CQM51L 24881331 IC50 = 63.9 nM T51191 C4KH8F 24881332 IC50 = 57.4 nM T51191 C1KA3V 24881333 IC50 = 216 nM T51191 C47APB 24881402 IC50 = 112 nM T51191 CSN8W1 24881403 IC50 = 167 nM T51191 C1UQ3K 24881404 IC50 = 47.5 nM T51191 C51TMH 24881405 IC50 = 77.4 nM T51191 C9EZI7 24881406 IC50 = 64.4 nM T51191 C6P3HS 24881407 IC50 = 124 nM T51191 CZ3TU1 24881464 IC50 = 146 nM T51191 CDI49N 24881465 IC50 = 124 nM T51191 CQGP87 24881466 IC50 = 116 nM T51191 CS1MH8 24888322 IC50 = 29000 nM T51191 CC0R9O 24938735 IC50 = 9.5 nM T51191 CF03HD 24948905 IC50 = 1740 nM T51191 CHP8O6 24948906 IC50 = 56.7 nM T51191 C1KRT8 24948907 IC50 = 1940 nM T51191 CKY2P8 24948908 IC50 = 147 nM T51191 C25CFI 24948909 IC50 = 1050 nM T51191 CWQ04Z 24948910 IC50 = 131 nM T51191 CM9I3X 24951310 IC50 = 133 nM T51191 CX1YF8 24951311 IC50 = 1690 nM T51191 CV10XU 24951312 IC50 = 238 nM T51191 CD6KV0 24951313 IC50 = 2980 nM T51191 CQY9Z0 24951314 IC50 = 93 nM T51191 CV8EF6 25032862 IC50 = 13 nM T51191 C35POS 25065102 IC50 >= 50 nM T51191 C62CND 25065309 IC50 >= 50 nM T51191 CNQ9O6 25065932 IC50 >= 50 nM T51191 CYC81K 25066135 IC50 >= 50 nM T51191 CZO9K3 25066136 IC50 >= 50 nM T51191 CH1Q5J 25066137 IC50 >= 50 nM T51191 CXD04I 25066140 IC50 = 500 nM T51191 CDF80L 25066350 IC50 = 500 nM T51191 CCKR19 25066353 IC50 >= 50 nM T51191 CX69SY 25066355 IC50 = 1930 nM T51191 CF8VP4 25066356 IC50 = 1570 nM T51191 CS9XH7 25066547 IC50 = 1540 nM T51191 C46AGN 25066548 IC50 = 207 nM T51191 CJF2M7 25066549 IC50 = 793 nM T51191 C7ZN2W 25118059 IC50 = 2.1 nM T51191 C4I1CJ 25155417 IC50 = 72 nM T51191 C72PBH 25155955 IC50 = 740 nM T51191 CB4E2J 25155956 IC50 = 71 nM T51191 CP4C5Y 25157071 IC50 = 470 nM T51191 CO14XG 25195084 IC50 = 140 nM T51191 C6BDX3 25207860 IC50 = 189000 nM T51191 CCD5M7 25227504 IC50 = 158 nM T51191 CK0D5S 25227505 IC50 = 382 nM T51191 CN97JP 25227508 IC50 = 268 nM T51191 CW8R1B 25227513 IC50 = 425 nM T51191 CE0NV4 25257993 IC50 = 4.39 nM T51191 C43BHY 25269097 IC50 = 54 nM T51191 CJ1RQ7 42598706 IC50 = 5160 nM T51191 C2LES7 42599455 IC50 = 3.1 nM T51191 C2KO0F 42599456 IC50 = 2.5 nM T51191 C1UAO7 42601485 IC50 = 14 nM T51191 CU23PG 42611301 IC50 = 5 nM T51191 CW1G2R 42611390 IC50 = 40 nM T51191 C62QFJ 42611486 IC50 = 70 nM T51191 CQ37HN 42612743 IC50 = 3.38 nM T51191 CX1UT9 42612744 IC50 = 825.2 nM T51191 CXK4C1 42618298 IC50 = 5 nM T51191 CQB20M 42630929 IC50 = 1700 nM T51191 CN93YB 42630930 IC50 > 5000 nM T51191 CH7RW1 42630932 IC50 = 450 nM T51191 CC8B0M 42630933 IC50 > 5000 nM T51191 CDT65Y 42631047 IC50 > 5000 nM T51191 CH69CQ 42631048 IC50 = 1200 nM T51191 C2NF6U 42632370 IC50 = 320 nM T51191 C2EA1T 42632371 IC50 = 310 nM T51191 C69LCN 42632491 IC50 = 1200 nM T51191 C9B8VR 42632614 IC50 > 5000 nM T51191 CB79DG 42637299 IC50 = 3600 nM T51191 CP36KB 42637300 IC50 > 100000 nM T51191 CI8J6H 42637372 IC50 = 530 nM T51191 C5RYO0 42637373 IC50 > 100000 nM T51191 CJ0CG5 42638004 IC50 = 99000 nM T51191 C8X0TG 42638005 IC50 = 830 nM T51191 CO57GS 44138033 IC50 = 15800 nM T51191 CQ2VD5 44219634 IC50 = 164 nM T51191 CY0QB9 44253226 IC50 = 270 nM T51191 CZ8R1N 44253780 IC50 = 192 nM T51191 C7G5CO 44359547 IC50 = 890 nM T51191 CIT7A9 44359548 IC50 = 41000 nM T51191 CUM0Q6 44359555 IC50 = 5900 nM T51191 CP92JV 44359673 IC50 > 100000 nM T51191 CQ7J2G 44359674 IC50 = 7800 nM T51191 CGK71T 44359675 IC50 = 11000 nM T51191 C2V4DN 44359681 IC50 = 1400 nM T51191 CX31TB 44359788 IC50 = 19000 nM T51191 CQ5Y8G 44359800 IC50 > 100000 nM T51191 CL82CH 44359814 IC50 > 100000 nM T51191 C5YRC9 44431499 IC50 = 110000 nM T51191 CK2P0J 44443716 IC50 = 500 nM T51191 CQ1WD9 44443718 IC50 = 500 nM T51191 CNC51G 44447194 IC50 = 105 nM T51191 C5VP4D 44454144 IC50 = 360 nM T51191 CJ0L4C 44456965 IC50 = 170 nM T51191 C74LTB 44506448 IC50 = 33 nM T51191 CPDE25 44507029 IC50 = 6300 nM T51191 C2UZ1P 44507247 IC50 = 560 nM T51191 CBL69N 44507542 IC50 = 20000 nM T51191 C7F8YJ 44543715 Ki = 125 nM T51191 CIO34V 44564642 Ki = 39 nM T51191 CG9OD1 44571302 IC50 = 520 nM T51191 C0ZX1A 44571330 IC50 = 5540 nM T51191 CY83MO 44571331 IC50 = 1810 nM T51191 CP6D1G 44571332 IC50 = 3470 nM T51191 CMA3R6 44574139 IC50 = 430 nM T51191 C5KLR7 44574177 IC50 > 30000 nM T51191 CFS49I 44574178 IC50 > 30000 nM T51191 CJ32DK 44574179 IC50 > 30000 nM T51191 CQOS28 44574180 IC50 = 469 nM T51191 CN96ZV 44574181 IC50 = 3750 nM T51191 CWJA85 44574206 IC50 > 30000 nM T51191 C46XHW 44574207 IC50 > 30000 nM T51191 C3RY9V 44574208 IC50 > 30000 nM T51191 CT7F0N 44589856 IC50 = 110 nM T51191 CA6Q9Y 44592060 IC50 = 13200 nM T51191 C5H8RA 44598536 IC50 = 290 nM T51191 CC2QV9 44623002 IC50 > 50000 nM T51191 CVJ51M 44623152 IC50 > 50000 nM T51191 C6TJ2G 44623153 IC50 > 50000 nM T51191 C8I7GL 44818075 IC50 > 1000 nM T51191 C42SJP 45141750 IC50 = 239 nM T51191 CLE9U5 45141751 IC50 = 589 nM T51191 CSM1O6 45271073 IC50 = 1100 nM T51191 C2M4GV 46179732 IC50 = 27.5 nM T51191 CS75CD 46179779 IC50 = 25.1 nM T51191 C39YKM 46179780 IC50 = 48.2 nM T51191 C0CKE5 46180624 IC50 > 30000 nM T51191 C7GYH0 46180758 IC50 = 60 nM T51191 C27IKH 46180759 IC50 = 24.6 nM T51191 CSC1Y9 46180760 IC50 = 28.5 nM T51191 C70FSJ 46180763 IC50 = 27.8 nM T51191 C0W8DB 46187719 IC50 = 1630 nM T51191 CV7D4Z 46187885 IC50 = 920 nM T51191 C53ZSX 46187886 IC50 = 8150 nM T51191 CEV52J 46187887 IC50 = 1580 nM T51191 CSC70G 46187888 IC50 = 8560 nM T51191 C7SC8A 46187889 IC50 = 2790 nM T51191 CQLG06 46187890 IC50 = 4530 nM T51191 CVGN05 46187891 IC50 = 7320 nM T51191 CF29IN 46188075 IC50 = 1050 nM T51191 COWJ59 46190552 IC50 > 10000 nM T51191 C8YO4W 46190553 IC50 > 10000 nM T51191 CEX48K 46190554 IC50 > 10000 nM T51191 C6J9DI 46190555 IC50 = 7690 nM T51191 C53RNX 46190556 IC50 > 10000 nM T51191 CPS37G 46190557 IC50 = 8520 nM T51191 C2MOT0 46190609 IC50 = 9230 nM T51191 CJ8OT2 46190610 IC50 > 10000 nM T51191 CX93ZQ 46190753 IC50 = 1170 nM T51191 C85WSJ 46190754 IC50 > 10000 nM T51191 C9VEX6 46190755 IC50 = 5190 nM T51191 C6O5AD 46190756 IC50 = 230 nM T51191 C7F8AM 46190820 IC50 = 7930 nM T51191 C8JY0S 46190821 IC50 = 1250 nM T51191 CUCK61 46190822 IC50 = 1560 nM T51191 CXQ51Y 46190823 IC50 = 2780 nM T51191 CR0G9O 46190824 IC50 = 390 nM T51191 CDP80X 46190825 IC50 = 510 nM T51191 C3ETP2 46190826 IC50 = 6260 nM T51191 CD57RJ 46197798 IC50 = 31 nM T51191 CR04HA 46197799 IC50 = 48 nM T51191 CQ83FI 46203315 IC50 = 730 nM T51191 CK8YL5 46203316 IC50 = 680 nM T51191 C1YB9P 46203618 IC50 = 3850 nM T51191 C4I5DH 46203619 IC50 > 10000 nM T51191 C43KVC 46203620 IC50 = 6290 nM T51191 CY7ER9 46203621 IC50 > 10000 nM T51191 CW13ZY 46203622 IC50 > 10000 nM T51191 CND31M 46203623 IC50 = 5190 nM T51191 C1RX2K 46203949 IC50 = 3160 nM T51191 CZJ86R 46203950 IC50 = 2870 nM T51191 CNA07J 46203951 IC50 = 2570 nM T51191 CQ69AM 46205433 IC50 = 165 nM T51191 CQTI31 46881225 IC50 > 30000 nM T51191 CVDH51 46887335 IC50 = 10000 nM T51191 CPS5F8 46887435 IC50 = 21000 nM T51191 CJ26EB 46887436 IC50 = 10000 nM T51191 CZP2B8 46887476 IC50 = 3800 nM T51191 C25DSY 46887918 IC50 = 179 nM T51191 C93CLK 46887919 IC50 = 11400 nM T51191 CPSI47 46890583 Ki = 12 nM T51191 C90NYX 46896338 IC50 = 250 nM T51191 CAT34L 46906643 IC50 = 90400 nM T51191 C4V7PG 46907052 IC50 = 10400 nM T51191 CMQ3R0 46907054 IC50 = 16500 nM T51191 C2PC1Z 46907160 IC50 = 96300 nM T51191 C1HV6U 46907409 IC50 = 20 nM T51191 CXH64A 46918825 IC50 = 25118.86 nM T51191 C6GY9I 46934544 IC50 = 18900 nM T51191 C3OD2Y 46934546 IC50 = 36200 nM T51191 CH61CW 47187185 IC50 > 1000 nM T51191 CL7PS1 49831258 IC50 > 50000 nM T51191 CI5L2P 49846123 IC50 = 563.7 nM T51191 C4DL0M 49847150 IC50 = 128 nM T51191 CC7Y9U 49850262 IC50 = 360 nM T51191 C50PXU 49855444 IC50 > 50000 nM T51191 C6POK9 49856931 IC50 = 14 nM T51191 C52ABG 50942502 IC50 = 290 nM T51191 CPQ0F7 50991199 IC50 = 29 nM T51191 COA5W3 51051073 IC50 = 82 nM T51191 C8U2AI 51180076 IC50 > 1000 nM T51191 CV76KB 51357270 IC50 = 72 nM T51191 CE43FC 53249967 IC50 > 30000 nM T51191 C7MO2J 53325871 IC50 = 26.5 nM T51191 CG84JS 53325976 IC50 = 800 nM T51191 CVM4Q3 53357987 IC50 = 3900 nM T51191 C78GKN 53361474 IC50 = 1000 nM T51191 CNB63X 53361475 IC50 = 780 nM T51191 CQ43VH 53363518 Ki = 8.6 nM T51191 C6Y2EV 53374826 IC50 = 6360 nM T51191 C9U7GF 53464577 IC50 = 4 nM T51191 C4EYP7 53464578 IC50 = 361.8 nM T51191 C0WNH9 53464579 IC50 = 199.4 nM T51191 C4MQ3U 53464638 IC50 = 2.3 nM T51191 CJ53ZV 53464639 IC50 = 381.1 nM T51191 CN9RH2 53464770 IC50 = 189.3 nM T51191 C5A7MU 54613496 IC50 = 34.1 nM T51191 CJ1G6K 56591671 IC50 = 670 nM T51191 CIO96M 56659403 IC50 > 100000 nM T51191 C7R9TZ 56663191 IC50 = 0.9 nM T51191 CL18NI 56666337 IC50 > 100000 nM T51191 C9LC5Y 56673234 IC50 > 100000 nM T51191 CWH5N4 56673261 IC50 > 100000 nM T51191 C2ML5S 56837168 IC50 = 20.4 nM T51191 CCW89V 56932477 IC50 = 1.11 nM T51191 CZ25SN 56935695 IC50 > 30000 nM T51191 CP4EL2 57328394 IC50 = 28000 nM T51191 CW02FD 57393108 IC50 = 740 nM T51191 CX0I2Z 57396604 IC50 = 880 nM T51191 CB8N4P 57400091 IC50 = 800 nM T51191 C5CRJ1 57412107 IC50 = 320 nM T51191 COG4Q8 57412108 IC50 = 190 nM T51191 C4LI0D 57521296 IC50 = 31000 nM T51191 CXFJ46 57550498 IC50 = 2700 nM T51191 CWT6O0 57723146 IC50 = 140 nM T51191 CA5Q6O 58147189 IC50 > 50000 nM T51191 C4DYC0 58147224 IC50 > 50000 nM T51191 CMP04X 58147302 IC50 > 50000 nM T51191 CLD40J 58465708 IC50 = 39000 nM T51191 C1MB4Q 59323957 IC50 > 30000 nM T51191 CK6LX0 59454220 IC50 = 220 nM T51191 C2SDN1 59454252 IC50 = 270 nM T51191 CO6A2S 59585196 IC50 = 710000 nM T51191 CLN20W 60143424 IC50 = 39.6 nM T51191 CEF0C3 60143425 IC50 = 43.6 nM T51191 CRNZ07 60145504 IC50 = 38.2 nM T51191 C31TUG 60145641 IC50 = 44.1 nM T51191 CG6M7H 60145642 IC50 = 3.9 nM T51191 C8XKG0 60145643 IC50 = 45.2 nM T51191 CC72HW 60145644 IC50 = 46.6 nM T51191 CBHR24 60145645 IC50 = 40.7 nM T51191 CS85AJ 60145783 IC50 = 48.1 nM T51191 C8SZ7X 60145784 IC50 = 5.2 nM T51191 CIP62A 60145785 IC50 = 45.5 nM T51191 CZPN39 60145786 IC50 = 48.5 nM T51191 CGX45C 60145787 IC50 = 40.3 nM T51191 CPZ5Q3 60148646 IC50 > 50000 nM T51191 C8ZL3J 60148690 IC50 > 50000 nM T51191 CK5N4E 60148693 IC50 = 43000 nM T51191 CB7X2E 60151224 IC50 = 45 nM T51191 CY05OU 60151225 IC50 = 328 nM T51191 CWO8H0 60152596 IC50 = 2710 nM T51191 CXW14A 60164619 IC50 = 12589.25 nM T51191 C5F0OQ 62706003 IC50 = 210 nM T51191 CQAM69 62706004 IC50 = 3200 nM T51191 C6CK5L 62706005 IC50 = 2400 nM T51191 C08BWT 62706006 IC50 = 10000 nM T51191 COTB68 62706167 IC50 = 830 nM T51191 CM0LI9 62706168 IC50 = 750 nM T51191 C5I8OL 62706169 IC50 = 77000 nM T51191 CW48QK 62706170 IC50 = 1000 nM T51191 CIQ52T 62706171 IC50 = 350 nM T51191 C8V2NC 62706321 IC50 = 1000 nM T51191 CBN3L0 69950064 Ki > 19000 nM T51191 C6RFQ8 70676597 IC50 > 20000 nM T51191 CD0YC8 70681968 IC50 = 4870 nM T51191 CM62BN 70682297 IC50 = 1580 nM T51191 CH2OA7 70684090 IC50 = 4990 nM T51191 C60XID 70684091 IC50 = 1150 nM T51191 C8L6YP 70686231 IC50 = 570 nM T51191 CGJK81 70686232 IC50 = 1150 nM T51191 CWF4E8 70688346 IC50 = 5020 nM T51191 CTE30H 70690378 IC50 = 6520 nM T51191 C7VF1B 70692849 Ki = 33 nM T51191 C28UMB 70693708 IC50 = 32 nM T51191 C1JO8E 70694590 IC50 = 2670 nM T51191 CWJ39I 70694591 IC50 = 2360 nM T51191 CE67KO 70695508 IC50 = 3300 nM T51191 C3DW5T 70696631 IC50 = 2170 nM T51191 CD5O7B 70696632 IC50 = 550 nM T51191 CQY1I6 70789579 Ki > 19000 nM T51191 CQ2E6U 71142135 IC50 = 3680 nM T51191 C8NZA0 71449818 IC50 = 72000 nM T51191 C63AHI 71449819 IC50 = 79000 nM T51191 C3J9QZ 71453454 IC50 = 1200 nM T51191 C57ATO 71455172 IC50 = 2000 nM T51191 C6B2HJ 71456958 IC50 = 300 nM T51191 CM9A3I 71458827 IC50 = 370 nM T51191 C72DJO 71465631 IC50 = 62 nM T51191 C0CX7P 71476624 Ki = 0.22 nM T51191 C6QPH1 71476625 Ki = 0.04 nM T51191 C3JLD4 71476626 Ki = 0.12 nM T51191 C3OH6T 71476627 Ki = 0.51 nM T51191 C0LWJ6 71520631 IC50 = 1392 nM T51191 CO28HI 71520716 IC50 = 944 nM T51191 CVA5Q7 71520717 IC50 = 881 nM T51191 C89SWX 71527724 IC50 > 30000 nM T51191 C6S5JQ 71527847 IC50 = 321.6 nM T51191 C6KBD4 71534512 IC50 = 1900 nM T51191 CT51EW 71534810 IC50 = 60 nM T51191 C7QN3O 71534812 IC50 = 15 nM T51191 C8M3HU 71537640 IC50 = 2230 nM T51191 C2QML7 71537641 IC50 = 37 nM T51191 CU0ZE6 71537928 IC50 = 78 nM T51191 CH9FS7 71537929 IC50 = 601 nM T51191 CTW95A 71537931 IC50 = 48 nM T51191 C3C0RO 71538475 IC50 = 70 nM T51191 CIA28E 71538746 IC50 = 67 nM T51191 CFCV26 71538748 IC50 = 2540 nM T51191 CY2T1Q 71538749 IC50 = 1770 nM T51191 C4A6VJ 71538750 IC50 = 68 nM T51191 CG72NC 71538751 IC50 = 168 nM T51191 C7RUE6 71540743 IC50 = 32100 nM T51191 C9LA4F 71540744 IC50 = 3880 nM T51191 C0EK5J 71540745 IC50 = 30800 nM T51191 C80HZX 71540746 IC50 = 224 nM T51191 C5UZQ0 71540747 IC50 = 25100 nM T51191 C4G5US 71540862 IC50 = 3270 nM T51191 CDW81Y 71574856 IC50 = 16790 nM T51191 CX01BJ 71574948 IC50 = 341 nM T51191 CO8YU7 71574949 IC50 = 1610 nM T51191 CBZ5S9 71583103 IC50 = 26000 nM T51191 C3PSJ9 71583105 IC50 = 29000 nM T51191 C21GHR 71624738 IC50 = 1200 nM T51191 CU65GH 71655059 IC50 = 657.7 nM T51191 CPS58L 71655136 IC50 = 468.3 nM T51191 CFW7Q9 71655137 IC50 = 414.2 nM T51191 C9S0UB 71655138 IC50 = 467.2 nM T51191 CU27EV 71655139 IC50 = 600.1 nM T51191 CO8R1Z 71655216 IC50 = 463.3 nM T51191 C0W6EK 71655283 IC50 = 881.8 nM T51191 C7HG0K 71655802 IC50 = 1790 nM T51191 CPJ4V7 71680913 IC50 = 9000 nM T51191 C9X8KM 71680914 IC50 = 20000 nM T51191 C4W2MA 71680915 IC50 = 11000 nM T51191 C3KO9V 71680916 IC50 = 30000 nM T51191 CN4X5O 71680917 IC50 > 33000 nM T51191 CWAM13 71680918 IC50 > 33000 nM T51191 CI9G3B 71681069 IC50 = 4800 nM T51191 CFUC24 71722010 IC50 = 111.2 nM T51191 CEG67K 71723449 IC50 = 1120 nM T51191 CTSK68 71811225 IC50 = 6450 nM T51191 C1K6OW 71811226 IC50 = 4000 nM T51191 CU3N9R 71811227 IC50 = 1610 nM T51191 CS2L4B 71811228 IC50 = 2210 nM T51191 CL4DT9 71811229 IC50 = 1220 nM T51191 CK6DB4 71811230 IC50 > 12000 nM T51191 CHR8V0 71811259 IC50 = 4810 nM T51191 CVL54T 71811261 IC50 > 10000 nM T51191 CZR93K 71811262 IC50 = 6880 nM T51191 CM8BE4 71811290 IC50 = 4780 nM T51191 C0MV3O 71811291 IC50 > 10000 nM T51191 C7UYD4 71811292 IC50 = 7480 nM T51191 C7XL3N 71811293 IC50 > 10000 nM T51191 C4HBC5 71811294 IC50 > 10000 nM T51191 CTA26S 71811295 IC50 = 5680 nM T51191 C9GHU8 71818097 IC50 = 111 nM T51191 CAW2Q1 71818098 IC50 = 81 nM T51191 CE89AK 71818242 IC50 = 580 nM T51191 C8M3IX 71818243 IC50 = 920 nM T51191 CKP5J7 71818244 IC50 = 440 nM T51191 CT7L6G 72163687 Ki = 0.25 nM T51191 CKE9D3 72163688 Ki = 0.23 nM T51191 CI9H6L 72164895 IC50 = 231 nM T51191 CS5UL7 72195322 IC50 = 397 nM T51191 CAC5Q7 72375561 IC50 = 1300 nM T51191 C3WQV2 72375562 IC50 = 20 nM T51191 CC1W6J 72375670 IC50 = 2100 nM T51191 CY8R0O 72696205 IC50 = 10390 nM T51191 C56QXM 72696206 IC50 = 53520 nM T51191 C0CM8Q 72696335 IC50 = 140 nM T51191 C73XOU 72734382 IC50 = 1150 nM T51191 CJR6C9 72734542 IC50 = 770 nM T51191 CV09DJ 72734543 IC50 = 3.5 nM T51191 CS6LW0 72946640 IC50 = 89 nM T51191 CXM37Z 72946641 IC50 = 142 nM T51191 CQA16N 72946833 IC50 = 143 nM T51191 CNR7Z2 72946834 IC50 = 689 nM T51191 C12JYS 72946835 IC50 = 238 nM T51191 C5Y9XH 72946836 IC50 = 110 nM T51191 CVZR94 72946837 IC50 = 5040 nM T51191 C8-AUG 72946838 IC50 = 956 nM T51191 CHQ39Y 72947043 IC50 = 143 nM T51191 CCST90 72947044 IC50 = 27 nM T51191 C7J3RH 72947045 IC50 = 93 nM T51191 CK10LZ 73292342 IC50 > 12000 nM T51191 CX3W1T 73333311 IC50 = 16000 nM T51191 CDG47J 73346009 IC50 > 20000 nM T51191 C6H7IJ 73346010 IC50 > 20000 nM T51191 CD0WU2 73346011 IC50 > 20000 nM T51191 COBJ19 73347538 IC50 = 1430 nM T51191 C92HFB 73349064 IC50 > 20000 nM T51191 C68LBO 73349131 IC50 = 21 nM T51191 CAS8E2 73352138 IC50 > 20000 nM T51191 C0C2QO 73353595 IC50 > 20000 nM T51191 C59WMZ 73353596 IC50 = 16700 nM T51191 C1UDF8 73353597 IC50 = 248 nM T51191 CUD02X 73355098 IC50 = 134 nM T51191 CXK86S 73355189 IC50 = 193 nM T51191 CD6L5K 73707349 IC50 = 1 nM T51191 C26KZD 73707535 IC50 = 6.9 nM T51191 CM1H3U 73707536 IC50 = 18.8 nM T51191 CH97TE 73707543 IC50 = 14.2 nM T51191 C2PWQ3 73707544 IC50 = 21 nM T51191 CEM5B6 73707545 IC50 = 6.3 nM T51191 CPQ43R 73707550 IC50 = 10.8 nM T51191 CJ1DA8 73774764 IC50 = 498.5 nM T51191 CQ3K6G 73776326 IC50 = 535.5 nM T51191 CC4L0G 73776327 IC50 = 432.1 nM T51191 CZB6G7 73776472 IC50 = 498.1 nM T51191 CSRE84 73776614 IC50 = 457 nM T51191 C01FVX 73776616 IC50 = 413.6 nM T51191 C3UC9H 73891099 IC50 = 10000 nM T51191 CM6H9C 76324878 IC50 > 50000 nM T51191 CL4JQ3 76331862 IC50 = 4390 nM T51191 C08CPW 76335428 IC50 = 180 nM T51191 C7JQU3 76335755 IC50 = 5840 nM T51191 CKI74A 76853213 IC50 > 20000 nM T51191 CCR7L2 76853289 IC50 > 100000 nM T51191 CJ6Z0X 78324068 IC50 > 20000 nM T51191 C3U0KE 81689842 IC50 > 50000 nM T51191 CG5ZD9 86291495 IC50 = 8.2 nM T51191 C61VCD 86294741 IC50 = 400000 nM T51191 CBWV30 86294747 IC50 = 95000 nM T51191 C06YBD 86302594 IC50 = 9490 nM T51191 C3EM7H 86581004 IC50 = 20 nM T51191 C7UK3Y 86581005 IC50 = 93 nM T51191 CY64UM 86581152 IC50 = 18 nM T51191 CY5V7C 86581153 IC50 = 10 nM T51191 C1HE8I 86581432 IC50 = 100 nM T51191 CZM07I 86581434 IC50 = 22 nM T51191 C8ZQG9 86581435 IC50 = 25 nM T51191 C6M9PL 86765212 IC50 = 1160 nM T51191 CS5I4Y 87261507 IC50 = 160 nM T51191 CQ2LF5 88920533 IC50 > 10000 nM T51191 CP1NA9 89183138 IC50 = 156 nM T51191 CQS6C0 89183185 IC50 = 219 nM T51191 CWY3H6 90024758 IC50 > 1000 nM T51191 CSBC45 90024759 IC50 > 1000 nM T51191 CB73DR 90025023 IC50 > 1000 nM T51191 C5P3DT 90025027 IC50 > 1000 nM T51191 C9GB2A 90025255 IC50 > 1000 nM T51191 C5W0UY 90025331 IC50 > 1000 nM T51191 C7NHW6 90025915 IC50 > 1000 nM T51191 CRC9B5 90026100 IC50 > 1000 nM T51191 CR53ON 90026278 IC50 > 1000 nM T51191 CX2U6G 90063981 IC50 > 1000 nM T51191 CZB49Y 90063982 IC50 > 1000 nM T51191 C8RG2T 90064049 IC50 > 1000 nM T51191 C2YQM7 90064053 IC50 > 1000 nM T51191 C62GSL 90654859 IC50 = 791.2 nM T51191 CJH1S6 90654947 IC50 > 10000 nM T51191 C94IWR 90654948 IC50 > 10000 nM T51191 CSR56C 90655296 IC50 = 5610 nM T51191 CSDO81 90664458 Ki = 27 nM T51191 CAQL21 91667420 IC50 = 69.8 nM T51191 C5M9AK 91667421 IC50 = 20.77 nM T51191 CJO6T1 91810840 IC50 = 2200 nM T51191 CYJ12Q 91884636 IC50 = 78 nM T51191 C34WIG 92045024 IC50 > 100000 nM T51191 C9OC0F 101882265 IC50 = 109000 nM T51191 CDV40P 101882454 IC50 = 160 nM T51191 C2I8XR 101882814 Ki = 1400 nM T51191 CVE07R 101882857 IC50 = 2230 nM T51191 C63EWT 101882858 IC50 = 3290 nM T51191 C8KZB4 101883993 Ki = 900 nM T51191 C7Q6ID 101884982 IC50 = 33 nM T51191 CR46PQ 101884983 IC50 = 34 nM T51191 CRZ83C 101884989 IC50 = 171 nM T51191 CT7Z8F 102514716 IC50 > 10000 nM T51191 CS2UL0 117829456 IC50 = 170 nM T51191 C7L4OT 117829461 IC50 = 100 nM T51191 C50VUN 117829462 IC50 = 90 nM T51191 CH27PR 118613747 IC50 = 21 nM T51191 C0OX4M 118613748 IC50 = 1.1 nM T51191 CNF09H 118613750 IC50 = 150 nM T51191 C3ETI2 118613751 IC50 = 3.1 nM T51191 C9KZQ0 118613755 IC50 = 1.4 nM T51191 C30OPU 118613756 IC50 = 6.3 nM T51191 C46TFD 118613757 IC50 = 1.4 nM T51191 C1J5AG 118613783 IC50 = 1.7 nM T51191 C9T0ML 118613821 IC50 = 1.1 nM T51191 CSU52M 118656852 IC50 > 30000 nM T51191 CB6AJ9 118656853 IC50 > 30000 nM T51191 C45UYG 118709095 IC50 = 33000 nM T51191 C7QHE4 118712502 IC50 = 0.5 nM T51191 C8KSD6 118712503 IC50 = 0.9 nM T51191 C1JFZ7 118714371 IC50 = 2747 nM T51191 CXF0U3 118714375 IC50 = 558 nM T51191 C2M5OR 118714376 IC50 = 204 nM T51191 CY4GN9 118714377 IC50 = 226 nM T51191 CM5QT7 118719376 Ki = 1700 nM T51191 CPB7C3 118719377 Ki = 600 nM T51191 C09OGH 118719378 Ki = 400 nM T51191 CR5VC1 118719379 Ki = 800 nM T51191 C32LCM 118719380 Ki = 300 nM T51191 C8U6YR 118719381 Ki = 300 nM T51191 C9Y0HV 118719382 Ki = 300 nM T51191 CY0J4D 118719383 Ki = 300 nM T51191 CCYU59 118719817 IC50 = 12 nM T51191 CSC47W 118720522 IC50 = 864.5 nM T51191 CUI51W 118720529 IC50 = 64.8 nM T51191 CCGH73 118720703 IC50 = 16400 nM T51191 CMV2W9 118721625 IC50 = 28 nM T51191 CF5TO3 118721859 IC50 = 103 nM T51191 CK97TZ 118721860 IC50 = 13 nM T51191 CYV30O 118721861 IC50 = 14 nM T51191 C5WYI1 118721862 IC50 = 5 nM T51191 CSMW25 118721863 IC50 = 6640 nM T51191 C5B1KM 118721864 IC50 = 454 nM T51191 CG8LZ0 118721865 IC50 = 19400 nM T51191 CPCN23 118721866 IC50 = 14000 nM T51191 CM0A9U 118721867 IC50 = 10700 nM T51191 C8IAG9 118734664 IC50 = 10420 nM T51191 CJ6KL7 118734665 IC50 = 380 nM T51191 C2VQ5P 118734666 IC50 = 4910 nM T51191 CYF71E 118734667 IC50 = 190 nM T51191 CQC7H0 118734668 IC50 = 6730 nM T51191 CP27CN 118734669 IC50 = 270 nM T51191 CBIY72 118734670 IC50 > 20 ug.mL-1 T51191 C9C7UX 118734705 IC50 = 5410 nM T51191 C16OUT 118735146 IC50 = 530 nM T51191 CZRV81 118735147 IC50 = 560 nM T51191 CFE4D0 118735148 IC50 = 290 nM T51191 C97NHV 118735149 IC50 = 5930 nM T51191 CQ0FJ3 118735150 IC50 = 430 nM T51191 CD4J8E 118735151 IC50 = 150 nM T51191 C7UE8T 118735152 IC50 = 280 nM T51191 CS6WO5 118735153 IC50 = 4390 nM T51191 C4XZ3C 118735154 IC50 = 8370 nM T51191 CRL6V4 118735155 IC50 = 320 nM T51191 CI8G4X 118737400 IC50 = 1770 nM T51191 C2F8TQ 118737455 IC50 = 380.5 nM T51191 C1T6WZ 118738004 IC50 > 10000 nM T51191 CZ61KV 118753026 IC50 = 1500 nM T51191 CFI23Y 118753027 IC50 = 6000 nM T51191 C75LTK 118753189 IC50 = 27000 nM T51191 C8DVP1 118868599 Ki = 7244 nM T51191 C9G4LD 118868621 Ki = 234 nM T51191 CQT5I6 118868656 Ki = 6097 nM T51191 CE3PD1 118868670 Ki > 10000 nM T51191 C5L8QM 118884518 IC50 = 3340 nM T51191 CV0E3L 118884590 Ki = 484 nM T51191 CME8R7 118884591 Ki = 1356 nM T51191 C4XJ7F 118884592 Ki = 66.51 nM T51191 CP5TE9 118884676 Ki = 943 nM T51191 CVTL89 118884679 Ki = 370 nM T51191 CB84TO 121278998 IC50 > 50000 nM T51191 C9S5OK 121279020 IC50 > 50000 nM T51191 CL3M2F 121499152 IC50 = 168 nM T51191 C93JAV 122177622 IC50 = 255 nM T51191 C5HJ0C 122177623 IC50 > 10000 nM T51191 CSU97K 122177957 IC50 = 275 nM T51191 CR8WL1 122180003 IC50 > 10000 nM T51191 CW4K2U 122181880 IC50 = 349.5 nM T51191 CK63UH 122181881 IC50 = 655.4 nM T51191 C0H9WU 122181882 IC50 = 4.42 nM T51191 CR3TU6 122181883 IC50 = 471.8 nM T51191 C57VRL 122181884 IC50 = 1240 nM T51191 C9V6XI 122186483 IC50 = 270 nM T51191 CU74JP 122186484 IC50 = 180 nM T51191 C7M2EU 122186485 IC50 = 360 nM T51191 CCG1Z2 122186543 IC50 = 610 nM T51191 CI32QY 122186544 IC50 = 250 nM T51191 CBN3P1 122186553 IC50 = 192 nM T51191 CP83NA 122186554 IC50 = 94 nM T51191 CPN31F 122191258 IC50 > 5000 nM T51191 CL5WI0 122191259 IC50 > 5000 nM T51191 CRTN32 122191260 IC50 = 1050 nM T51191 C1ZRE6 122191261 IC50 > 5000 nM T51191 C97BGS 122191262 IC50 > 5000 nM T51191 C1GUZ3 122191263 IC50 > 5000 nM T51191 CJG60T 122191264 IC50 > 5000 nM T51191 C28JVO 122192004 IC50 = 36.6 nM T51191 CF2D8U 122192005 IC50 = 2740 nM T51191 CW1HK5 122195536 IC50 = 6.8 nM T51191 C5W8OZ 122376192 IC50 = 25.6 nM T51191 C3V5ND 122550211 IC50 = 386 nM T51191 C63EYP 122601008 IC50 > 3000 nM T51191 CCN03D 122601010 IC50 > 10000 nM T51191 CZC01M 122601076 IC50 > 3000 nM T51191 CZE35C 122648343 IC50 = 3.9 nM T51191 C54RNT 122648367 IC50 = 2.9 nM T51191 C1UVI7 122648600 IC50 = 11.46 nM T51191 CMX59K 122648648 IC50 = 2.62 nM T51191 CVZ64I 122648649 IC50 = 2.8 nM T51191 CJR97Y 123525532 IC50 > 1000 nM T51191 CVFI87 127025051 IC50 > 10000 nM T51191 CE4CI8 127025178 IC50 = 221 nM T51191 CM38EU 127025541 IC50 = 140 nM T51191 CY5T9P 127025646 IC50 > 3000 nM T51191 CKJ6L8 127025647 IC50 > 3000 nM T51191 C6D2IJ 127026516 IC50 = 165 nM T51191 C8BA3S 127027767 IC50 = 56 nM T51191 CG8NU7 127027995 IC50 = 72 nM T51191 CZ7C3D 127028030 IC50 = 3.3 nM T51191 CV07OM 127028943 IC50 = 68 nM T51191 CV9I8D 127030313 IC50 = 5200 nM T51191 CR0P1O 127031793 IC50 = 11800 nM T51191 C4GI0F 127037614 IC50 = 187 nM T51191 CSJ32V 127039213 IC50 = 154 nM T51191 CZ8A1F 127041696 IC50 = 29850 nM T51191 C5D2OJ 127044292 IC50 = 1450 nM T51191 C58KRZ 127044343 IC50 = 4730 nM T51191 C1TYS6 127044344 IC50 = 119 nM T51191 C3G0SM 127044498 IC50 = 1290 nM T51191 C5CP9M 127045259 IC50 = 6560 nM T51191 CB8HR2 129104138 IC50 > 50000 nM T51191 CCH65A 129104183 IC50 > 50000 nM T51191 CFH8Q4 129104227 IC50 > 50000 nM T51191 C6HM5P 129104349 IC50 > 50000 nM T51191 CZTF90 129104374 IC50 > 50000 nM T51191 CUJ2P5 129104402 IC50 > 50000 nM T51191 CY3I6X 129104426 IC50 > 50000 nM T51191 CGT6B0 130238385 Ki = 469 nM T51191 CMWV13 130238420 Ki = 310 nM T51191 C0GH4T 130238474 Ki = 70.8 nM T51191 C9ERM5 130238475 Ki = 768 nM T51191 C8IEV4 130258911 IC50 = 1870 nM T51191 CHVF85 132022730 IC50 > 100000 nM T51191 C6OXE3 132134663 IC50 = 49 nM T51191 CP8L7V 132137973 IC50 = 3103 nM T51191 C6X3HG 132145728 IC50 = 8610 nM T51191 C8O9DP 132157820 IC50 = 12500 nM T51191 C2N5JD 132279660 IC50 = 135 nM T51191 C4L6UZ 132547258 IC50 = 163 nM T51191 CGBR54 132547259 IC50 = 4050 nM T51191 CW4MP2 132547260 IC50 = 854 nM T51191 C1YO2Z 132547261 IC50 = 407 nM T51191 CU63DV 132569672 IC50 = 256 nM T51191 CIUZ08 132576538 IC50 = 439 nM T51191 CTE3A6 132576539 IC50 = 659 nM T51191 C87DPY 132576540 IC50 = 827 nM T51191 CG91UP 132576541 IC50 = 1788 nM T51191 CL2R5W 132576542 IC50 = 759 nM T51191 C5C2EQ 132576544 IC50 = 1294 nM T51191 CA5V0R 132576546 IC50 = 2915 nM T51191 C0Y2TP 132585192 IC50 = 66 nM T51191 C4KE3N 132938351 IC50 = 268 nM T51191 C4UAN3 134129876 IC50 = 294 nM T51191 C25EVA 134129883 IC50 = 302 nM T51191 CWRH43 134129994 IC50 = 232 nM T51191 CK2TM6 134130010 IC50 = 2060 nM T51191 CYW6H1 134130165 IC50 = 32 nM T51191 CQ7SN8 134131102 IC50 = 929 nM T51191 CQO23I 134131456 IC50 = 209 nM T51191 CHZ8A3 134131564 IC50 = 1360 nM T51191 CN9DL4 134132030 IC50 > 10000 nM T51191 CX93QK 134135812 IC50 > 100000 nM T51191 CN8L9J 134136160 IC50 = 580000 nM T51191 C53UTO 134137062 IC50 = 1100 nM T51191 CSX58U 134139437 IC50 = 3330 nM T51191 C08YTI 134140697 IC50 = 15 nM T51191 C75NRQ 134141877 IC50 > 100000 nM T51191 C62SVR 134142119 IC50 > 100000 nM T51191 CLI48U 134143743 IC50 = 14100 nM T51191 CUA26W 134143927 IC50 = 58000 nM T51191 CWRJ15 134147087 IC50 > 100000 nM T51191 C8K0XJ 134147090 IC50 = 3370 nM T51191 CQ61SB 134150479 IC50 = 86500 nM T51191 CDX75O 134152551 IC50 = 15000 nM T51191 C2JV5X 134153768 IC50 > 100000 nM T51191 C2E8MV 134154228 IC50 = 11.48 nM T51191 C38DIF 134156853 IC50 = 180000 nM T51191 C4FLQ5 134157355 IC50 > 100000 nM T51191 C1UP3S 134157845 IC50 = 2250 nM T51191 C0X1HQ 134224487 IC50 = 570 nM T51191 CZV43J 134283792 IC50 = 18000 nM T51191 C62WXO 134283796 IC50 = 51000 nM T51191 CO7K3N 134283799 IC50 = 4900 nM T51191 CBQ17L 134283800 IC50 = 36000 nM T51191 C1Y4TA 134283810 IC50 = 38000 nM T51191 CV2YF7 134283813 IC50 = 32000 nM T51191 C05FVT 134492522 IC50 > 10000 nM T51191 C52IBY 134823859 IC50 = 18000 nM T51191 CS1V6A 135367138 IC50 > 50000 nM T51191 CVO59N 135367789 IC50 > 50000 nM T51191 CDY18W 135407493 IC50 > 100000 nM T51191 CW2I4R 135412048 IC50 > 100000 nM T51191 C7U0AV 135412194 IC50 > 100000 nM T51191 CS54TL 135437514 IC50 = 67000 nM T51191 C36MUC 135441620 IC50 > 100000 nM T51191 CRB8M1 135444536 IC50 > 100000 nM T51191 CX5D6J 135446479 IC50 = 18900 nM T51191 C1TOK2 135449197 IC50 > 100000 nM T51191 CW25GL 135462117 IC50 > 100000 nM T51191 CCL28F 135473106 IC50 > 100000 nM T51191 CYA60G 135497781 IC50 > 100000 nM T51191 C01EZF 135567459 IC50 > 100000 nM T51191 CV3QP4 135886613 IC50 = 108 nM T51191 C8X5LO 135928012 Ki = 70 nM T51191 CI2YE8 135928628 IC50 > 100000 nM T51191 C50NIS 136025837 IC50 > 100000 nM T51191 C4OS0V 136025842 IC50 > 100000 nM T51191 CX7Z5B 136025843 IC50 > 100000 nM T51191 CB8EM9 136025984 IC50 > 100000 nM T51191 C49MUG 136025986 IC50 > 100000 nM T51191 C0OLS8 136030779 IC50 = 65000 nM T51191 CIA7R4 136030780 IC50 = 76000 nM T51191 C24LKN 136030781 IC50 > 100000 nM T51191 CH7Y3C 136086920 IC50 > 100000 nM T51191 C3VDL5 136086921 IC50 > 100000 nM T51191 C9GOB5 136086922 IC50 = 69300 nM T51191 CE3ZL7 136086923 IC50 > 100000 nM T51191 CJZ5F3 136086924 IC50 > 100000 nM T51191 CT19ND 136110961 IC50 = 110 nM T51191 CY9U0E 136173089 IC50 = 110 nM T51191 C19VDS 136237971 IC50 = 19200 nM T51191 CBS97C 136239447 IC50 = 85 nM T51191 CT2MI6 136239448 IC50 = 44 nM T51191 CE2F9G 136244081 IC50 = 56 nM T51191 C9CH7S 136244085 IC50 = 104 nM T51191 C5J2AX 136244086 IC50 = 82 nM T51191 C46CYT 136244087 IC50 = 425 nM T51191 CXY1L5 136244088 IC50 = 538 nM T51191 CILG36 136286746 IC50 = 117 nM T51191 C39WRP 136286747 IC50 > 20000 nM T51191 C7ZX5O 136286761 IC50 = 3860 nM T51191 C9SV6G 136645392 IC50 > 20000 nM T51191 CANQ56 136645396 IC50 > 20000 nM T51191 C9TGH1 136645397 IC50 > 20000 nM T51191 C1F7JV 136645401 IC50 > 20000 nM T51191 C32LNQ 136645404 IC50 = 14600 nM T51191 C4W0IE 136645405 IC50 > 20000 nM T51191 CMIU28 136645406 IC50 > 20000 nM T51191 C3K2WL 136645410 IC50 = 11400 nM T51191 CC1D0X 136645415 IC50 = 17500 nM T51191 C02RIK 136645417 IC50 > 20000 nM T51191 C8CT0Z 136645422 IC50 = 1110 nM T51191 CAWT82 136645431 IC50 = 1110 nM T51191 CBZ8Q1 136645433 IC50 > 20000 nM T51191 C21EJD 136645435 IC50 > 20000 nM T51191 C1KTV3 136645436 IC50 > 20000 nM T51191 CK1B9W 136645438 IC50 = 2550 nM T51191 C6QOP7 136645441 IC50 = 4800 nM T51191 CMZ71T 136645444 IC50 > 20000 nM T51191 CL47WS 136645445 IC50 = 799 nM T51191 C64BZR 136645447 IC50 > 20000 nM T51191 C7X1UL 136645449 IC50 = 1260 nM T51191 CI9ZO7 136645454 IC50 = 5190 nM T51191 CA3I8S 136645455 IC50 > 20000 nM T51191 CRN16W 136645457 IC50 = 1310 nM T51191 CGQ92L 136645458 IC50 = 6970 nM T51191 CO5DN2 136645462 IC50 = 4640 nM T51191 CRPN39 136645466 IC50 = 3720 nM T51191 CL5X3G 136645467 IC50 = 17500 nM T51191 C48HNY 136959539 IC50 = 1850 nM T51191 C1P8ZW 136959550 IC50 = 490 nM T51191 CKU95F 136966187 IC50 = 712 nM T51191 CFRG19 136985286 IC50 > 20000 nM T51191 CE7F4O 136985287 IC50 = 166 nM T51191 CFPT21 136985288 IC50 = 1940 nM T51191 CBH5Y0 136985291 IC50 = 2030 nM T51191 CDAK28 136985292 IC50 = 341 nM T51191 CQ9XW7 136985295 IC50 > 20000 nM T51191 C1M6NW 136985296 IC50 > 20000 nM T51191 CJOA28 136985302 IC50 = 4390 nM T51191 CE6QK0 137125258 IC50 = 160 nM T51191 CAW80Q 137125259 IC50 = 130 nM T51191 CP5NM4 137125260 IC50 = 280 nM T51191 C5CKZ8 137125261 IC50 = 180 nM T51191 C1ROQ9 137125262 IC50 = 290 nM T51191 CL29YN 137125263 IC50 = 180 nM T51191 C5OY8K 137125264 IC50 = 150 nM T51191 C0YGR6 137125265 IC50 = 240 nM T51191 CMYG96 137125266 IC50 = 340 nM T51191 CI78CK 137125267 IC50 = 230 nM T51191 CD62KP 137125268 IC50 = 400 nM T51191 CE8NM5 137125269 IC50 = 430 nM T51191 CANS59 137136982 IC50 > 20000 nM T51191 C5AE3Q 137283418 IC50 > 20000 nM T51191 C5QIX1 137289788 IC50 = 1860 nM T51191 C5X0YR 137289866 IC50 = 335 nM T51191 CU70ZB 137289868 IC50 > 20000 nM T51191 CV6AN7 137289892 IC50 > 20000 nM T51191 CB14CI 137289900 IC50 > 20000 nM T51191 CLY69S 137289946 IC50 > 20000 nM T51191 CC5HA4 137290225 IC50 > 20000 nM T51191 C4RBC7 137290234 IC50 > 20000 nM T51191 CKJ6Q4 137290238 IC50 > 20000 nM T51191 CR53GQ 137290273 IC50 = 490 nM T51191 C8DYG6 137290344 IC50 > 20000 nM T51191 C9G3JB 137292402 IC50 = 89 nM T51191 C6MXL3 137292504 IC50 = 6430 nM T51191 CAZ49O 137300702 IC50 = 1870 nM T51191 CGE0J6 137300703 IC50 = 13900 nM T51191 CDU43L 137300704 IC50 = 9830 nM T51191 CK0QG6 137300705 IC50 > 20000 nM T51191 C91IPL 137300706 IC50 > 20000 nM T51191 C5UYP8 137300707 IC50 > 20000 nM T51191 CHSG63 137300708 IC50 = 2250 nM T51191 CX57MR 137300709 IC50 = 14100 nM T51191 C54KGS 137300710 IC50 = 432 nM T51191 CQD07Z 137300711 IC50 > 20000 nM T51191 C3I1CB 137300712 IC50 > 20000 nM T51191 C9LP2B 137353123 IC50 = 1100 nM T51191 CNKJ27 137353141 IC50 = 1300 nM T51191 CAW4X1 137353146 IC50 = 3000 nM T51191 CAPH58 137353182 IC50 = 3200 nM T51191 CWM6Z2 137376574 Ki = 995 nM T51191 C3LUJ0 137487429 IC50 = 5300 nM T51191 CA5OY1 137628667 IC50 = 179 nM T51191 C67EFJ 137628684 IC50 = 0.61 nM T51191 CHL7E8 137631592 IC50 = 320 nM T51191 CJ7P1U 137631803 IC50 = 441 nM T51191 C1N8TU 137632249 Ki = 3195 nM T51191 C84MIY 137633138 IC50 = 337 nM T51191 CW8G1H 137633768 IC50 = 193.5 nM T51191 C82QCH 137633786 IC50 = 209.35 nM T51191 C73PDL 137634086 IC50 = 75 nM T51191 C1V8QE 137634156 IC50 = 6309.57 nM T51191 CZ1FK2 137635119 IC50 = 28.04 nM T51191 C6JVG9 137635398 IC50 = 5.8 nM T51191 CAWZ25 137635575 IC50 = 0.53 nM T51191 COF8J3 137635708 IC50 = 21.2 nM T51191 C2KS3O 137635975 IC50 = 3130 nM T51191 CK1S0F 137637029 IC50 = 3.9 nM T51191 CEI0W2 137637915 IC50 = 2500 nM T51191 CTUL07 137638741 IC50 = 0.9 nM T51191 CX8Q4R 137638837 Ki = 313 nM T51191 CDWG31 137638917 IC50 = 209 nM T51191 CUG0C9 137639328 IC50 > 10000 nM T51191 CJBF37 137639551 IC50 = 287.59 nM T51191 C3CD6L 137639796 IC50 = 2319.76 nM T51191 C06BYV 137640258 IC50 = 283.3 nM T51191 C19GDO 137640291 IC50 = 59.5 nM T51191 CS50ET 137641009 IC50 = 1340 nM T51191 C4OEC3 137641520 IC50 = 1300 nM T51191 C5JUR2 137641533 IC50 = 1040 nM T51191 C1PRH5 137642860 IC50 = 61 nM T51191 C37BJQ 137642900 IC50 = 194 nM T51191 CJOS87 137643760 IC50 = 223 nM T51191 C7DLO4 137644089 IC50 = 490 nM T51191 CCBN61 137645084 IC50 = 311 nM T51191 C8GNS5 137645287 IC50 = 3215.9 nM T51191 C8WPM4 137645400 IC50 = 1650 nM T51191 CX3E0H 137645675 IC50 = 121.3 nM T51191 C5REZ8 137645689 IC50 > 20000 nM T51191 CA0V2Q 137647353 IC50 = 146 nM T51191 CM65KH 137647813 IC50 = 0.18 nM T51191 CO7H5A 137648171 IC50 = 179 nM T51191 CN3I9X 137648982 IC50 = 111 nM T51191 C0PGD9 137649617 IC50 = 314 nM T51191 CGK2M9 137649620 IC50 = 90 nM T51191 CM15FY 137649624 IC50 > 10000 nM T51191 CEP9R0 137651700 IC50 = 970 nM T51191 CFLX25 137652000 IC50 = 2380 nM T51191 C8NHK9 137652359 IC50 > 5000 nM T51191 C5FHD3 137652442 IC50 = 20300 nM T51191 CMP7G0 137652638 IC50 = 121 nM T51191 CZI5S2 137653293 IC50 = 170 nM T51191 C3QX5N 137653295 IC50 = 332.1 nM T51191 CXZ5J3 137654094 IC50 = 84 nM T51191 CIW9C6 137654210 Ki = 5205 nM T51191 C3FEM8 137654512 IC50 = 1640 nM T51191 CCR5B3 137654793 IC50 = 47 nM T51191 C1SBN5 137654946 IC50 = 1408.14 nM T51191 C71ZNJ 137656226 IC50 > 10000 nM T51191 CVG9T3 137656290 IC50 = 26 nM T51191 C0NR1V 137656498 IC50 = 1460 nM T51191 CRP0T2 137656638 IC50 = 1270 nM T51191 C0EQI2 137656898 IC50 = 296 nM T51191 C76OGQ 137656942 IC50 = 24000 nM T51191 CY8A2I 137656945 IC50 = 88.77 nM T51191 C5BM7T 137657586 IC50 = 908 nM T51191 C97QUM 137657678 IC50 = 179 nM T51191 C21XDS 137657845 IC50 = 3500 nM T51191 CPJL30 137659007 IC50 = 217 nM T51191 C9D7NR 137659196 IC50 = 199.3 nM T51191 CFGW13 137659898 IC50 = 128 nM T51191 C6XWP9 137659968 IC50 = 385.51 nM T51191 CM0OE5 137660128 IC50 = 1120 nM T51191 CLWU57 137660171 IC50 = 191.3 nM T51191 CEJI95 137661885 IC50 = 69 nM T51191 CEF18M 137661927 IC50 > 5000 nM T51191 CAQ62X 137701235 Ki = 23 nM T51191 CXV84M 138377596 IC50 = 120 nM T51191 CIWG23 138393067 IC50 = 910 nM T51191 C7EM3I 138393071 IC50 = 568 nM T51191 C4NFS3 138393072 IC50 = 420.5 nM T51191 CA3C4O 138454792 IC50 = 3 nM T51191 CN2UH1 139303146 IC50 = 13.26 nM T51191 CN4M1E 139325532 IC50 = 2100 nM T51191 C9EBI4 139325820 IC50 = 8400 nM T51191 CP73QO 141504704 IC50 = 1260 nM T51191 C13JZX 141522811 IC50 = 47100 nM T51191 CHS9N0 141728829 IC50 = 730 nM T51191 C9H8PX 141728841 IC50 = 130 nM T51191 CBV2K5 141728842 IC50 = 190 nM T51191 C2HF9A 141728845 IC50 = 430 nM T51191 C4RGY1 141728867 IC50 = 1400 nM T51191 C7XI0V 141764754 IC50 = 3.6 nM T51191 CO6C7N 142489312 IC50 = 2800 nM T51191 C7B3JK 142489313 IC50 = 4800 nM T51191 CGT08I 142489314 IC50 = 1800 nM T51191 CF7K4G 142489316 IC50 = 2700 nM T51191 CM6LR2 142489318 IC50 = 2500 nM T51191 C42DBC 142489319 IC50 = 3000 nM T51191 CH5Y8E 142489322 IC50 = 1100 nM T51191 C5MN8W 142489323 IC50 = 2000 nM T51191 CFYC82 142489328 IC50 = 1200 nM T51191 C4DKW7 142489330 IC50 = 7800 nM T51191 CDS81U 142489335 IC50 = 630 nM T51191 CMY8W1 142489337 IC50 > 10000 nM T51191 CD5E9S 142489342 IC50 = 2000 nM T51191 C65LBI 142489344 IC50 = 3400 nM T51191 CX0E9B 142505968 IC50 = 14100 nM T51191 CBJC50 142505992 IC50 = 18190 nM T51191 C7N8LV 142506025 IC50 = 3247 nM T51191 CKBF56 142506033 IC50 = 1231 nM T51191 CGNQ74 142506189 IC50 = 7173 nM T51191 CP5HF8 142506225 IC50 = 25480 nM T51191 CF5CB6 144562551 IC50 > 1000 nM T51191 C0CRK4 144562558 IC50 > 1000 nM T51191 C5I0NG 144562573 IC50 > 1000 nM T51191 CDI1U5 144562574 IC50 > 1000 nM T51191 CDA28I 145949712 IC50 = 23 nM T51191 CXJ0Y4 145949850 IC50 = 20 nM T51191 C1EF9X 145950102 IC50 = 114 nM T51191 CRKM19 145950884 IC50 = 6.8 nM T51191 CV3QO5 145951170 IC50 = 999.6 nM T51191 CRSM78 145952088 IC50 = 32900 nM T51191 CFE4G6 145952135 IC50 = 263 nM T51191 CEC68O 145952295 IC50 = 4900 nM T51191 CKG98W 145953085 IC50 > 100000 nM T51191 CL0XT8 145954248 IC50 = 25 nM T51191 CM53ZB 145954785 IC50 = 10800 nM T51191 CNB9E6 145955015 IC50 = 4200 nM T51191 CGP9X1 145955496 IC50 = 232 nM T51191 CJ03TU 145957740 IC50 = 413 nM T51191 CBNG29 145957781 IC50 = 32 nM T51191 C3L8IE 145958641 IC50 = 1704 nM T51191 C8SI2G 145958925 IC50 > 10000 nM T51191 CO05IK 145959360 IC50 = 132 nM T51191 C9IV1C 145959866 IC50 = 33.1 nM T51191 CK1XI0 145960971 IC50 > 10000 nM T51191 C1X5EO 145962694 IC50 = 33 nM T51191 C29PAL 145963897 IC50 = 29000 nM T51191 CJ47DY 145964043 IC50 > 100000 nM T51191 C3PWD4 145964064 IC50 = 1950 nM T51191 CEX67F 145964240 IC50 = 47000 nM T51191 CEDK05 145964533 IC50 = 5500 nM T51191 CDO47P 145964554 IC50 = 40000 nM T51191 CDY56B 145964885 IC50 = 424 nM T51191 CB51JU 145965019 IC50 > 100000 nM T51191 CW6UM7 145965159 IC50 = 3100 nM T51191 C9XLE7 145966296 IC50 > 100000 nM T51191 CM6KY1 145966543 IC50 > 100000 nM T51191 CJAE67 145966594 IC50 = 7250 nM T51191 CTUF34 145966712 IC50 = 380 nM T51191 CTRI57 145966861 IC50 > 100000 nM T51191 CUD38A 145967089 IC50 = 2700 nM T51191 C19POY 145967140 IC50 = 5140 nM T51191 C93JKN 145967593 IC50 = 1974 nM T51191 CD82XB 145967610 IC50 = 135 nM T51191 C7OG1D 145967698 IC50 = 635 nM T51191 C5RPQ9 145967832 IC50 = 47 nM T51191 CI1ZD2 145967851 IC50 = 2883 nM T51191 CR59HK 145967905 IC50 = 883 nM T51191 C95SNQ 145967968 IC50 = 919 nM T51191 CES7W6 145968087 IC50 = 1503 nM T51191 CSO4I7 145968364 IC50 > 5000 nM T51191 CSJ81Y 145968726 IC50 = 1800 nM T51191 CG0S9U 145968824 IC50 = 763 nM T51191 CIA79M 145968985 IC50 = 114 nM T51191 C27YHM 145969456 IC50 = 40 nM T51191 CV53YN 145969651 IC50 = 391 nM T51191 C0K6XS 145969789 IC50 = 76 nM T51191 CZ80EP 145969996 IC50 = 1216 nM T51191 C79YOL 145970069 IC50 > 100000 nM T51191 CFL68X 145970091 IC50 > 100000 nM T51191 C7TSV2 145970161 IC50 = 1835 nM T51191 CG5OK8 145970171 IC50 = 42 nM T51191 C3FQ0V 145970292 IC50 = 11200 nM T51191 C8FXH4 145970309 IC50 = 99000 nM T51191 CBR60K 145970453 IC50 = 362 nM T51191 C0E2UO 145970598 IC50 = 17 nM T51191 CI43DY 145970786 IC50 = 1770 nM T51191 C7K1AJ 145971681 IC50 = 7472 nM T51191 CA0F3X 145972521 IC50 > 1000 nM T51191 CW0T7A 145973234 IC50 = 5740 nM T51191 CO51JK 145973368 IC50 = 98.8 nM T51191 C4HTO2 145973543 IC50 = 2140 nM T51191 CSR50O 145973656 IC50 = 70400 nM T51191 CFP2R3 145973876 IC50 > 100000 nM T51191 CVM0Z3 145974125 IC50 > 100000 nM T51191 CLCU89 145974270 IC50 = 5400 nM T51191 C8YEJ9 145974425 IC50 = 5110 nM T51191 CUJE21 145974558 IC50 > 10000 nM T51191 CY1G2F 145974565 IC50 = 491 nM T51191 C5YJO8 145974667 IC50 = 58000 nM T51191 CZL05M 145975187 IC50 > 100000 nM T51191 CE8I5V 145975869 IC50 = 4800 nM T51191 C6Y9QH 145975913 IC50 = 69000 nM T51191 CU65BZ 145976000 IC50 > 100000 nM T51191 C86GXV 145976671 IC50 = 13000 nM T51191 CMUA94 145976675 IC50 = 7270 nM T51191 CN6UO4 145977003 IC50 = 11600 nM T51191 CKAQ67 145977127 IC50 = 3030 nM T51191 C78XNS 145977336 IC50 > 100000 nM T51191 CLY4Z5 145977632 IC50 = 240 nM T51191 CP53JS 145977717 IC50 = 16.6 nM T51191 C3QYB8 145978561 IC50 > 100000 nM T51191 COR40V 145978805 IC50 = 2100 nM T51191 C7X4LZ 145978932 IC50 = 900 nM T51191 C0UG8S 145980171 IC50 = 390 nM T51191 CIM41N 145980574 IC50 = 410 nM T51191 CMB08D 145981960 IC50 = 147 nM T51191 CMY73B 145983639 IC50 = 6300 nM T51191 CWD0A9 145983712 Ki = 3.1 nM T51191 CB24HO 145985400 IC50 = 470 nM T51191 C56MWZ 145986208 Ki = 130 nM T51191 C1WH7V 145986586 IC50 > 5000 nM T51191 CS79CE 145986632 IC50 = 327 nM T51191 CRX8H1 145987492 IC50 = 41 nM T51191 CPAX89 145987732 IC50 = 40 nM T51191 CJ1M7T 145987832 IC50 = 6.6 nM T51191 CV3S8R 145988041 IC50 = 3230 nM T51191 C82CIN 145988785 IC50 > 30000 nM T51191 CJ8DO3 145989487 IC50 = 549 nM T51191 C68VKC 145993051 IC50 = 370 nM T51191 C1W6CF 145994016 IC50 = 12000 nM T51191 C0YXS8 147254231 IC50 = 4618 nM T51191 C48EXH 148289288 IC50 = 9.25 nM T51191 CN71OS 149405396 IC50 = 13620 nM T51191 CWG10H 151364732 IC50 = 97 nM T51191 C6I7OZ 152636346 IC50 = 85 nM T51191 C7LM4U 153534003 IC50 = 251 nM T51191 CP1V9H 153534004 IC50 = 105 nM T51191 C9FIY4 153534005 IC50 = 58 nM T51191 CVT63S 153534008 IC50 = 170 nM T51191 C7JFY3 154068925 IC50 > 1000 nM T51191 C0KW3O 155511274 IC50 = 174.6 nM T51191 C0LH8C 155511921 IC50 = 282 nM T51191 CB8RS9 155512087 IC50 > 25000 nM T51191 CV2MG0 155512401 IC50 = 81 nM T51191 CT4VS3 155512474 IC50 = 150 nM T51191 CQ5BL7 155512551 IC50 > 50000 nM T51191 C7VKU2 155513116 IC50 = 139 nM T51191 CHLO32 155513171 IC50 = 1300 nM T51191 C5WUJ6 155513192 IC50 = 112 nM T51191 CE4H7I 155513471 IC50 > 50000 nM T51191 CCDH73 155514314 IC50 = 5400 nM T51191 C6BV9W 155514532 IC50 = 1240 nM T51191 CW3VT9 155514603 IC50 > 50000 nM T51191 CZ84WI 155515284 IC50 > 50000 nM T51191 CWEZ05 155515488 IC50 = 2.46 nM T51191 CUKG21 155515602 IC50 > 50000 nM T51191 CYJ53T 155515864 IC50 = 8100 nM T51191 C1K2XN 155516139 IC50 = 4942 nM T51191 CRS8L2 155516458 IC50 > 1000 nM T51191 CA1J3N 155517086 IC50 = 249 nM T51191 CL72ME 155517175 IC50 = 49.5 nM T51191 C7G0XM 155517418 IC50 = 4100 nM T51191 CY54TU 155518062 IC50 > 30000 nM T51191 CEH2N5 155518106 IC50 = 277 nM T51191 C58ZNC 155518327 IC50 = 7.42 nM T51191 CCDU61 155518496 IC50 = 205 nM T51191 C5ZQ3R 155519423 IC50 > 1000 nM T51191 CDY5H6 155519645 IC50 = 4910 nM T51191 C34FXY 155520399 IC50 = 9835 nM T51191 CAD10S 155520741 IC50 > 10000 nM T51191 CAZ3S7 155521187 IC50 = 16000 nM T51191 CZ75FW 155521272 IC50 = 203 nM T51191 CG4F2U 155521283 IC50 = 144 nM T51191 C82PHV 155521822 IC50 = 3060 nM T51191 C6DVZ9 155521965 IC50 = 5030 nM T51191 C0KJ1Z 155522601 IC50 > 10000 nM T51191 C63KJW 155523399 IC50 > 1000 nM T51191 CG84WO 155523907 IC50 = 1493 nM T51191 CU5RZ1 155524034 IC50 = 665 nM T51191 CJ3E4G 155524660 IC50 = 6660 nM T51191 CYB97D 155525236 IC50 > 1000 nM T51191 C8DM2Y 155525412 IC50 > 1000 nM T51191 CI24AD 155525662 IC50 = 4214 nM T51191 CN7B1T 155525782 IC50 > 100000 nM T51191 CG1K0O 155526247 IC50 > 10000 nM T51191 COD92I 155526258 IC50 = 3500 nM T51191 C63NOC 155527045 IC50 = 662 nM T51191 CEM0A3 155527290 IC50 = 3222 nM T51191 CW2H5R 155527295 IC50 = 485 nM T51191 C71UNO 155527385 Ki = 70 nM T51191 CQK19H 155527955 IC50 = 786 nM T51191 C20FJM 155528257 IC50 > 1000 nM T51191 CHR4K5 155528532 IC50 > 100000 nM T51191 CZ70PO 155529066 IC50 > 50000 nM T51191 C49NGT 155529137 IC50 > 50000 nM T51191 C9L6OC 155529247 IC50 = 3.4 nM T51191 C94BFW 155529690 IC50 = 5950 nM T51191 C74OTA 155529983 IC50 = 1746 nM T51191 CU0C7W 155530254 IC50 = 500 nM T51191 CZMC49 155530597 IC50 = 24.5 nM T51191 C8AZI6 155530932 IC50 = 7316 nM T51191 CZG79N 155531159 IC50 = 474.1 nM T51191 CN3W5J 155531452 IC50 > 50000 nM T51191 CUC3P1 155531533 IC50 = 1600 nM T51191 CK2UY4 155531957 IC50 > 50000 nM T51191 CDJ0W3 155532052 IC50 = 1080 nM T51191 CZO38U 155532084 IC50 = 1885 nM T51191 CBCJ50 155532192 IC50 > 1000 nM T51191 C3HDI1 155532640 IC50 = 18.49 nM T51191 CD8ZV7 155532950 IC50 = 1820 nM T51191 CIZ46A 155533876 IC50 = 26000 nM T51191 C0T8AS 155533910 IC50 = 926 nM T51191 CPE68B 155534222 IC50 = 7943.28 nM T51191 C4ST9U 155534232 IC50 > 1000 nM T51191 C5FLH0 155535184 IC50 > 1000 nM T51191 C91UNV 155535585 IC50 = 140 nM T51191 C81KIF 155537008 IC50 = 160 nM T51191 C2JH0S 155537112 IC50 = 283 nM T51191 CQV6H0 155537405 IC50 = 8071 nM T51191 C5FRG0 155537455 IC50 = 172 nM T51191 CTF98X 155537473 IC50 = 420 nM T51191 CAG9P4 155537573 IC50 > 50000 nM T51191 C1PFV7 155538765 IC50 = 1817 nM T51191 CLD19W 155539311 IC50 = 1190 nM T51191 CU6V4Q 155539319 IC50 > 50000 nM T51191 CM5UN4 155539714 IC50 = 1366 nM T51191 CBO78Z 155540097 IC50 = 950 nM T51191 C6U0FM 155540189 IC50 = 14000 nM T51191 C6LQT1 155540719 IC50 > 5000 nM T51191 CKN07B 155541358 IC50 = 1267 nM T51191 C7B5NU 155541992 IC50 = 5380 nM T51191 C4T9YC 155542195 IC50 > 100000 nM T51191 CP4L1F 155544459 IC50 = 45000 nM T51191 CNM3P1 155544603 IC50 > 10000 nM T51191 CXR86J 155545078 IC50 > 50000 nM T51191 CCV9J0 155545380 IC50 = 21 nM T51191 C2UN1K 155545446 IC50 = 136 nM T51191 C1JSY3 155545907 IC50 = 135 nM T51191 C8DQ7U 155546022 IC50 = 107.5 nM T51191 CE1D7Q 155546207 IC50 > 100000 nM T51191 CF2O4J 155546325 IC50 > 50000 nM T51191 CK45LA 155546486 IC50 = 7943.28 nM T51191 C3HB0U 155546555 IC50 = 1995.26 nM T51191 CS3GO2 155546558 IC50 = 850 nM T51191 C0AU1L 155546632 IC50 > 50000 nM T51191 C8LT4A 155546691 IC50 = 67.48 nM T51191 CP3Q7I 155547009 IC50 = 8100 nM T51191 CHD0I6 155547367 IC50 = 2440 nM T51191 C1D4PI 155547606 Ki = 150 nM T51191 CTFU61 155549051 IC50 = 610 nM T51191 C90FBZ 155549087 IC50 > 50000 nM T51191 CE0YL6 155549538 IC50 = 200 nM T51191 CO6ID4 155550122 IC50 = 1000 nM T51191 CV4QP6 155550492 IC50 > 1000 nM T51191 C4Z5JX 155550827 IC50 = 50000 nM T51191 CA03BO 155551057 IC50 = 3162.28 nM T51191 C3JQ1N 155551780 IC50 = 668 nM T51191 C05ZVG 155552130 IC50 = 8320 nM T51191 CV4Y5B 155552792 IC50 = 1100 nM T51191 CXT8F1 155552802 IC50 = 12930 nM T51191 CH8L1V 155554197 IC50 = 860 nM T51191 CGDF76 155554360 IC50 = 24000 nM T51191 CC56ED 155554844 IC50 = 21 nM T51191 CXGR50 155555191 IC50 = 880 nM T51191 C8ZD2Y 155555330 IC50 = 4200 nM T51191 CF2H3O 155555451 IC50 = 489 nM T51191 CM7FN8 155555499 IC50 = 160 nM T51191 CFW90N 155555562 IC50 = 1.6 nM T51191 C8FZN4 155555652 IC50 > 1000 nM T51191 C7QTU1 155555957 IC50 > 50000 nM T51191 CIN57Q 155556138 IC50 = 1130 nM T51191 C6IL1E 155557199 IC50 = 278.6 nM T51191 CEX5I7 155557262 IC50 > 1000 nM T51191 CNM71L 155557418 IC50 = 579.3 nM T51191 C8AUB0 155558567 IC50 = 75 nM T51191 CK3B2T 155558642 IC50 = 3700 nM T51191 CPD50Q 155559583 IC50 = 3400 nM T51191 C26QOJ 155559606 IC50 > 1000 nM T51191 CC62UI 155559872 IC50 = 1810 nM T51191 CT31YW 155560779 IC50 = 7000 nM T51191 C13TBU 155560878 IC50 > 1000 nM T51191 CW50YA 155561265 IC50 = 1298 nM T51191 CH0Z1P 155561539 IC50 = 352 nM T51191 CJ4KO7 155562145 IC50 = 441.3 nM T51191 CGL24S 155562249 IC50 > 50000 nM T51191 CSJ23C 155562809 IC50 = 994 nM T51191 CM0DS1 155562992 IC50 > 1000 nM T51191 CBJ03Y 155563284 IC50 = 819 nM T51191 CXEQ27 155563524 IC50 = 1400 nM T51191 CXWU93 155563558 IC50 = 180 nM T51191 CX23YB 155564400 IC50 = 95.51 nM T51191 CR85ZW 155564587 IC50 = 1900 nM T51191 CPNA06 155564750 IC50 > 50000 nM T51191 C87JXN 155564870 IC50 = 6309.57 nM T51191 CG65CR 155565674 IC50 = 50000 nM T51191 CD05RS 155566122 IC50 > 50000 nM T51191 C4A0RK 155566461 IC50 > 50000 nM T51191 CP1MH4 155566833 IC50 = 8300 nM T51191 C04CGS 155567444 IC50 > 50000 nM T51191 CDT3W1 155567506 IC50 > 1000 nM T51191 CS03PJ 155568350 IC50 > 50000 nM T51191 CF2X0U 155568767 IC50 = 530 nM T51191 CW5XB4 155569484 IC50 = 147 nM T51191 C3BAZ5 24861442 IC50 = 12.7 nM T51191 D00GBB 11449246 Ki = 44 nM T51191 D00HXX 56650312 IC50 = 9700 nM T51191 D00KFF 9882812 IC50 = 1400 nM T51191 D00SEE 11379392 IC50 = 1300 nM T51191 D01AVS 25065930 IC50 = 500 nM T51191 D01FYB 23648267 IC50 = 2000 nM T51191 D01TSM 46887380 IC50 = 3800 nM T51191 D01YBR 44591988 IC50 = 27700 nM T51191 D02NWS 279980 Ki = 430 nM T51191 D02TQA 15986508 IC50 = 1860 nM T51191 D03QOD 239512 IC50 = 6600 nM T51191 D03TNE 25065710 IC50 = 500 nM T51191 D03TQD 25065713 IC50 = 500 nM T51191 D04KQF 6675804 Ki = 42 nM T51191 D04UVL 1133083 IC50 = 6980 nM T51191 D05OVV 11993691 IC50 = 2000 nM T51191 D05RWU 46887334 IC50 = 800 nM T51191 D06IWR 46887438 IC50 = 1300 nM T51191 D07BMT 46887378 IC50 = 3900 nM T51191 D07MYE 5355635 IC50 = 457 nM T51191 D07WSB 46887381 IC50 = 3100 nM T51191 D07YZZ 5173 Ki = 29 nM T51191 D08USK 46887437 IC50 = 13000 nM T51191 D08YLO 46830345 IC50 = 1400 nM T51191 D09RKA 72946782 IC50 = 0.112 nM T51191 D09SVH 25065929 IC50 = 500 nM T51191 D0A4KW 46830327 IC50 = 39 nM T51191 D0AK8Q 42632368 IC50 = 820 nM T51191 D0B3ZM 11436024 IC50 = 2220 nM T51191 D0D2US 25065931 IC50 = 500 nM T51191 D0E0TA 44454650 IC50 = 200 nM T51191 D0E9DD 16095101 Ki = 50 nM T51191 D0FI2F 25065925 IC50 = 500 nM T51191 D0G6DH 16661454 IC50 = 870 nM T51191 D0H4SC 46887439 IC50 = 600 nM T51191 D0H4YW 3611 Ki = 15.44 nM T51191 D0I2KC 46830328 IC50 = 43 nM T51191 D0K3MR 22915475 IC50 = 720 nM T51191 D0K7QR 45269423 IC50 = 590 nM T51191 D0M1ZI 16095112 Ki = 3000 nM T51191 D0M9LJ 44454415 IC50 = 900 nM T51191 D0MD7H 44454143 IC50 = 27 nM T51191 D0N9AK 44138031 IC50 = 11000 nM T51191 D0Q2GM 44454416 IC50 = 390 nM T51191 D0Q4LX 46887475 IC50 = 10000 nM T51191 D0Q5DI 71462653 Ki = 1250 nM T51191 D0Q5MC 24753719 IC50 = 31000 nM T51191 D0Q9PO 16095114 Ki = 10 nM T51191 D0T0SK 44138032 IC50 = 2670 nM T51191 D0T4JQ 264 IC50 = 12000 nM T51191 D0U8FC 759408 IC50 = 3100 nM T51191 D0W1PV 6918328 Ki = 0.12 nM T51191 D0W2PX 46887379 IC50 = 140 nM T51191 D0W9BH 15986510 IC50 = 330 nM T51191 D0X4VO 44359538 IC50 = 26000 nM T51191 D0XZ9Q 11149404 IC50 = 754 nM T51191 D0Y4SD 46887333 IC50 = 390 nM T51191 D0YO6M 785232 IC50 = 900 nM T51191 D0Z8PX 24757913 IC50 = 18.65 nM T92687 D01XNB 4594 IC50 = 250 nM T92687 D02DPA 2756 IC50 = 820 nM T92687 D0T6XX 4679 IC50 = 1000 nM T92687 D02THB 3081087 IC50 = 18000 nM T92687 C2KJI7 3883 IC50 = 398.11 nM T92687 C93BJO 5039 IC50 = 40 nM T92687 CL86ZR 72171 IC50 = 130000 nM T92687 C0K7OY 108137 IC50 = 65 nM T92687 C0V2PL 119157 IC50 = 700 nM T92687 C8A5QG 126974 IC50 = 1258.93 nM T92687 CS1W8P 126981 IC50 = 1000 nM T92687 CPZ9O5 134982 IC50 = 8080 nM T92687 C4PS8O 474505 IC50 = 2100 nM T92687 C18OEH 474509 IC50 = 600 nM T92687 C2W4JU 474510 IC50 = 800 nM T92687 CY70UT 474511 IC50 = 11000 nM T92687 CYQ34E 474513 IC50 = 200 nM T92687 CWS4F5 536278 IC50 = 1500 nM T92687 CQ79JG 3763607 IC50 = 40000 nM T92687 CV72KD 3780371 IC50 = 35000 nM T92687 CXE80F 7176102 IC50 = 20000 nM T92687 C9EM6K 7176110 IC50 = 60000 nM T92687 CM0UY5 7176114 IC50 = 33000 nM T92687 C09XMW 7176116 IC50 = 53000 nM T92687 CW45OL 9795949 IC50 = 4800 nM T92687 C8ZOW0 9796998 IC50 > 100000 nM T92687 CRMV29 9797594 IC50 = 17000 nM T92687 CR6Q0B 9798310 IC50 = 7200 nM T92687 CD84ZU 9798780 IC50 > 100000 nM T92687 CLAB14 9817871 IC50 = 8200 nM T92687 C1DV8G 9840636 IC50 = 72000 nM T92687 CR9KX3 9860166 IC50 = 530 nM T92687 C87GHA 9861877 IC50 = 14000 nM T92687 CG1SM3 9905717 IC50 = 5700 nM T92687 CY1Q7U 9925182 IC50 = 170 nM T92687 CM81WF 9927582 IC50 = 4800 nM T92687 C6U7QL 9969937 IC50 = 180 nM T92687 CPW49I 10109886 IC50 = 280 nM T92687 CM03ID 10133649 IC50 = 210 nM T92687 CTDN59 10134275 IC50 = 350 nM T92687 C57SPG 10136947 IC50 = 340 nM T92687 CW84KJ 10154608 IC50 = 250 nM T92687 CI8S7Q 10155379 IC50 = 270 nM T92687 CBGA43 10156387 IC50 = 170 nM T92687 CUVC78 10249325 IC50 = 24000 nM T92687 CHC07A 10269336 IC50 = 320 nM T92687 C25VYZ 10270162 IC50 = 80 nM T92687 C62JWA 10271847 IC50 = 110 nM T92687 C9ERN3 10293942 IC50 = 260 nM T92687 C57GMA 10386097 IC50 = 590 nM T92687 CQO04P 10526412 IC50 = 400 nM T92687 C54BAH 10549567 IC50 = 460 nM T92687 CD4HE3 10693875 IC50 = 1700 nM T92687 CGH09O 10716562 IC50 = 16600 nM T92687 C8GH6C 10788603 IC50 = 59000 nM T92687 CPZX36 10838303 IC50 = 1900 nM T92687 C24KHY 11269080 IC50 = 31622.78 nM T92687 CDFB43 11743300 IC50 = 16000 nM T92687 CEC10K 11795090 IC50 = 26000 nM T92687 C5DA3O 11795895 IC50 = 450 nM T92687 CG93NT 12041550 IC50 = 150 nM T92687 CRP72O 12399957 IC50 = 9000 nM T92687 C5HOD8 13338270 IC50 = 64 nM T92687 CCF4H7 13392898 IC50 = 23000 nM T92687 CX76WT 13392914 IC50 = 15000 nM T92687 CY5H0I 13392932 IC50 = 32000 nM T92687 COWS24 13537479 IC50 = 4300 nM T92687 CGLI79 13656363 IC50 = 600 nM T92687 C2O8DQ 13754158 IC50 = 13500 nM T92687 C2DT0M 13754159 IC50 = 4400 nM T92687 C86VRE 13754160 IC50 = 3200 nM T92687 CIJG42 13754162 IC50 = 2100 nM T92687 CJ34BV 13754165 IC50 = 1600 nM T92687 CF74WR 13754168 IC50 = 120000 nM T92687 C9AR7Z 13900248 IC50 = 400 nM T92687 CG3C2E 13900258 IC50 = 310 nM T92687 C9Q5GT 13900267 IC50 = 1460 nM T92687 CHWA94 14064679 IC50 = 24000 nM T92687 C31GLW 14064680 IC50 = 7400 nM T92687 CP3M8Z 14064681 IC50 = 7900 nM T92687 C8FZ5U 14064682 IC50 = 12000 nM T92687 CLV72Q 14064683 IC50 > 100000 nM T92687 CT47SM 14064684 IC50 = 700 nM T92687 CLZ68E 14064685 IC50 = 2000 nM T92687 CIO5A1 14064686 IC50 = 3900 nM T92687 C6QEG1 14064687 IC50 = 2600 nM T92687 CS24CK 14064688 IC50 = 9300 nM T92687 C3P4IV 14064689 IC50 > 100000 nM T92687 CX2OH1 14064690 IC50 = 25000 nM T92687 C03MHN 14064691 IC50 = 24000 nM T92687 CI7KQ2 14064692 IC50 > 100000 nM T92687 C7EZ8F 14064693 IC50 > 100000 nM T92687 CO05RP 14064694 IC50 > 100000 nM T92687 CZ20IW 14064695 IC50 = 4200 nM T92687 C3QP1W 14064696 IC50 = 5400 nM T92687 C89TAN 14064697 IC50 = 5300 nM T92687 C6UHA7 14064698 IC50 > 100000 nM T92687 CJV16H 14064699 IC50 = 8500 nM T92687 CG41PQ 14064700 IC50 = 800 nM T92687 CI3KR7 14064701 IC50 = 60000 nM T92687 COIJ05 14064702 IC50 = 6400 nM T92687 CWU3S0 14064703 IC50 = 1500 nM T92687 C2FHR5 14064704 IC50 = 700 nM T92687 CZ8R9K 14064705 IC50 = 16000 nM T92687 C42XNG 14064706 IC50 = 2700 nM T92687 CB3X5I 14146297 IC50 = 1500 nM T92687 CBR86X 14146299 IC50 = 420 nM T92687 C91CQU 14146301 IC50 = 230 nM T92687 CIVE53 14146303 IC50 = 340 nM T92687 CIH4G0 14146305 IC50 = 1800 nM T92687 C4F6DL 14146307 IC50 = 230 nM T92687 CBG1X0 14146309 IC50 = 3000 nM T92687 C21UAN 14146311 IC50 = 2000 nM T92687 CS0E5I 14146313 IC50 = 540 nM T92687 C92BLQ 14146315 IC50 = 1650 nM T92687 CNV6I8 14146317 IC50 = 310 nM T92687 C9SLE6 14146319 IC50 = 120 nM T92687 CW02CN 14146321 IC50 = 490 nM T92687 CBQ9F1 14146323 IC50 = 120 nM T92687 CJW31V 14146325 IC50 = 180 nM T92687 C50CJA 14146327 IC50 < 10000 nM T92687 C1HMJ5 14146329 IC50 = 50 nM T92687 C5Z6TN 14146331 IC50 = 80 nM T92687 CGZN76 14146335 IC50 = 310 nM T92687 CX26MI 14146337 IC50 = 370 nM T92687 CRZ8E4 14146339 IC50 = 3000 nM T92687 CU6C1H 14146351 IC50 = 50 nM T92687 CAJ34G 14146357 IC50 = 180 nM T92687 CX6SY9 14146371 IC50 = 250 nM T92687 CKI45L 14146373 IC50 = 530 nM T92687 CY65OU 14146375 IC50 = 260 nM T92687 C72MHQ 14146377 IC50 = 400 nM T92687 CVE2D7 14146379 IC50 = 150 nM T92687 CPUG47 14146381 IC50 = 140 nM T92687 CYKG52 14146384 IC50 = 130 nM T92687 CME7G0 14146386 IC50 = 430 nM T92687 C0JEU7 14146388 IC50 = 180 nM T92687 C9V3PS 14146390 IC50 = 30 nM T92687 CK0ZB1 14146392 IC50 = 160 nM T92687 CA63ZS 14146394 IC50 = 260 nM T92687 CFV2I6 14146397 IC50 = 250 nM T92687 C9ZEO2 14146401 IC50 = 1500 nM T92687 C4F5AE 14146403 IC50 = 2600 nM T92687 C0A2CP 14146405 IC50 = 1200 nM T92687 C59ZHY 14590341 IC50 = 3800 nM T92687 C0J4CI 14590350 IC50 = 14100 nM T92687 CBJE97 14590360 IC50 = 990 nM T92687 C0HK8T 14590362 IC50 = 17500 nM T92687 CT1P2Z 15163488 IC50 = 2511.89 nM T92687 CPS67D 15163489 IC50 = 1584.89 nM T92687 CT2O8F 15163490 IC50 = 501.19 nM T92687 CO6B1Y 15163491 IC50 = 630.96 nM T92687 CZY0X9 15163492 IC50 = 1000 nM T92687 C3KXD9 15163493 IC50 = 2511.89 nM T92687 CN90GC 15163494 IC50 = 794.33 nM T92687 C18YHB 15163495 IC50 = 5011.87 nM T92687 CPF38Y 15163496 IC50 = 19952.62 nM T92687 CC9L8W 15163497 IC50 = 7943.28 nM T92687 CQS19H 15163498 IC50 = 398.11 nM T92687 C38WMN 15163499 IC50 = 1258.93 nM T92687 CCHZ08 15163500 IC50 = 2511.89 nM T92687 CMLY48 15163501 IC50 = 15848.93 nM T92687 CH80ZD 15163502 IC50 = 3981.07 nM T92687 CH8I3Q 15163503 IC50 = 1584.89 nM T92687 CZ9D1S 15163504 IC50 = 7943.28 nM T92687 CGHI34 15163505 IC50 = 3162.28 nM T92687 CMD60R 15163510 IC50 = 63095.73 nM T92687 CPC2B7 15163511 IC50 = 2511.89 nM T92687 CT6J9K 15247229 IC50 = 1500 nM T92687 CL25VZ 15247231 IC50 = 1200 nM T92687 CD8CU1 15729210 IC50 = 28000 nM T92687 C8SOK4 15729211 IC50 = 1000 nM T92687 CN5PZ8 15729212 IC50 = 9800 nM T92687 C0ZR9X 15729213 IC50 = 7900 nM T92687 C26QMD 15729214 IC50 = 2900 nM T92687 C1J7KH 15729215 IC50 = 9100 nM T92687 C38CQZ 15729216 IC50 = 9000 nM T92687 CK6C3V 15729218 IC50 = 17000 nM T92687 CZ8ME4 15729222 IC50 = 11000 nM T92687 COQ70N 15729225 IC50 = 2000 nM T92687 CVJN41 15729229 IC50 = 7000 nM T92687 CU81YE 15729230 IC50 = 26000 nM T92687 CR4D9K 15729231 IC50 = 11000 nM T92687 C69MER 15729232 IC50 = 25000 nM T92687 CTYX02 15729234 IC50 = 6000 nM T92687 CN08PJ 15729236 IC50 = 7000 nM T92687 C3X9AR 15729238 IC50 = 1500 nM T92687 C5J4VC 15729239 IC50 = 4300 nM T92687 CRWU79 15729240 IC50 = 19000 nM T92687 C5H9KQ 15729242 IC50 = 1200 nM T92687 C9R4SD 15729243 IC50 = 1800 nM T92687 C9LK0T 15729244 IC50 = 3300 nM T92687 CEV0K3 15729245 IC50 = 1800 nM T92687 CIR29M 15729246 IC50 = 940 nM T92687 C5OYB7 15729247 IC50 = 1600 nM T92687 C47PZD 15729248 IC50 = 1600 nM T92687 C02KUW 15729249 IC50 = 7600 nM T92687 C78MJO 15729250 IC50 = 1000 nM T92687 C2F8NX 15729251 IC50 = 9000 nM T92687 CS7Y5V 15729252 IC50 = 1700 nM T92687 C3OW2J 15729253 IC50 = 960 nM T92687 CESQ51 15729254 IC50 = 700 nM T92687 CX7BM2 15729255 IC50 = 7400 nM T92687 C32NRG 15729256 IC50 = 2700 nM T92687 CC7O2L 15729257 IC50 = 6700 nM T92687 CMY47K 15729258 IC50 = 3100 nM T92687 C4L5FS 15729261 IC50 = 23800 nM T92687 CG3LC4 15729262 IC50 = 7600 nM T92687 CQ7R5V 15729263 IC50 = 590 nM T92687 CNH6V8 15729264 IC50 = 700 nM T92687 C7NA4J 19828026 IC50 = 14000 nM T92687 C7OP6G 19828037 IC50 = 6200 nM T92687 CEG6N1 19828052 IC50 = 8800 nM T92687 C1LPO4 20459002 IC50 = 130 nM T92687 C2D6IU 24854807 IC50 = 18000 nM T92687 C6XI3E 24854809 IC50 = 27000 nM T92687 CT7M9E 24854867 IC50 = 32000 nM T92687 CMFY87 44295365 IC50 = 10000 nM T92687 CRV2M0 44299282 IC50 = 98000 nM T92687 C5T0ZG 44299489 IC50 = 33000 nM T92687 C8PYE2 44299550 IC50 > 100000 nM T92687 C91MEQ 44299614 IC50 > 100000 nM T92687 CX8U5V 44327587 IC50 = 100000 nM T92687 C9MD8Q 44327856 IC50 = 3400 nM T92687 C0MT7Q 44327861 IC50 > 100000 nM T92687 CL9BW7 44327862 IC50 > 100000 nM T92687 CZ4ME9 44327865 IC50 = 80000 nM T92687 C09OMQ 44357574 IC50 = 442000 nM T92687 CZB76R 44367388 IC50 = 5300 nM T92687 C8Z7DM 44367389 IC50 > 50000 nM T92687 C8EIY0 44367454 IC50 = 21000 nM T92687 CJ0YI9 44367502 IC50 = 6000 nM T92687 CJQ82H 44367505 IC50 = 7000 nM T92687 CWBX89 44367624 IC50 = 10000 nM T92687 COV4P6 44367633 IC50 = 37000 nM T92687 CL6V0Y 44367634 IC50 = 6000 nM T92687 CUZ18J 44367635 IC50 = 2000 nM T92687 C2TO6H 44367644 IC50 = 11000 nM T92687 CUI1R3 44367655 IC50 = 9100 nM T92687 CB38UZ 44367657 IC50 = 27000 nM T92687 CRL67A 44367686 IC50 = 10000 nM T92687 CKFJ96 44367735 IC50 = 7000 nM T92687 CH1U0K 44367736 IC50 = 7000 nM T92687 C73JXF 44367748 IC50 = 1600 nM T92687 C7AQ2V 44367749 IC50 = 300 nM T92687 CWP95L 44367751 IC50 = 4200 nM T92687 C2J5FK 44367755 IC50 = 1300 nM T92687 CU7HE0 44367758 IC50 = 4000 nM T92687 CBK18J 44367761 IC50 = 5200 nM T92687 CVU9F6 44367772 IC50 = 1000 nM T92687 CF6RX8 44367773 IC50 = 14000 nM T92687 CHT9Z2 44367776 IC50 = 2300 nM T92687 CI9E5H 73348089 IC50 = 700 nM T92687 CH0DC8 73351177 IC50 = 700 nM T92687 C3M2TO 73355692 IC50 = 600 nM T92687 C72ILO 73357208 IC50 = 1100 nM T43760 C16ZSG 6439929 EC50 > 100000 nM T43760 C9G0MH 9803551 EC50 = 0.5 nM T43760 C3RI8T 9840880 EC50 = 110 nM T43760 CC64MT 9869395 Ki = 1380 nM T43760 CSN23P 9910192 EC50 = 8 nM T43760 C3Y0LD 10109471 EC50 = 15 nM T43760 C7GH9F 10161481 EC50 = 3.2 nM T43760 C1MX6V 10200104 EC50 = 0.08 nM T43760 CB1A0L 10224506 EC50 = 8 nM T43760 CJB2E3 10274474 EC50 = 0.5 nM T43760 CDI3H8 10298167 EC50 = 2.6 nM T43760 C1DB3O 11452211 EC50 = 4 nM T43760 C3WO0K 11455692 EC50 = 115 nM T43760 CW0GN2 11677766 EC50 = 3 nM T43760 CHTP62 15540528 EC50 = 23 nM T43760 C0CLM5 21018711 EC50 = 22 nM T43760 C3RP8C 22228616 EC50 = 1000 nM T43760 CEVG58 22228618 EC50 = 7 nM T43760 CDV16M 22228621 EC50 = 0.3 nM T43760 CT9CJ2 22228623 EC50 = 5.1 nM T43760 CP76IJ 22228633 EC50 = 210 nM T43760 CK08IC 44391337 EC50 = 1.2 nM T43760 CGQ95P 44391338 EC50 = 7.8 nM T43760 CDVK95 44391349 EC50 = 11 nM T43760 CRMJ60 44391353 EC50 = 0.2 nM T43760 CY8WC1 44391371 EC50 = 495 nM T43760 C8V4GJ 44391387 EC50 = 18 nM T43760 C0GU4F 44391396 EC50 = 15 nM T43760 C6JBK9 44391408 EC50 = 4 nM T43760 CFX12D 44391409 EC50 = 72 nM T43760 CKY54P 44391411 EC50 = 4 nM T43760 CX6W2B 44441125 EC50 = 1000 nM T43760 CXQ2U7 44441138 EC50 = 1000 nM T43760 CU73EN 44441145 EC50 = 0.06 nM T43760 C37VFI 44441147 EC50 = 70 nM T43760 CA9PL8 91663316 IC50 = 32400 nM T93580 D07XOD 2733079 IC50 = 30.1 nM T93580 D0E9JL 70690209 IC50 = 93300 nM T93580 CCI13U 11536910 IC50 = 7.2 nM T93580 CN8LG9 13171484 IC50 = 22.3 nM T93580 CXC3W5 20377108 IC50 = 23.5 nM T93580 C3PDB6 20377110 IC50 = 29.8 nM T93580 CI3Q2W 25125116 IC50 = 176 nM T93580 C5NER0 25125122 IC50 = 121 nM T93580 CGF7A0 25125458 IC50 = 52.3 nM T93580 CS1RD3 25125461 IC50 = 13.5 nM T93580 CJ4I7C 25125799 IC50 = 15.6 nM T93580 CM6EV5 70681820 IC50 = 14.4 nM T93580 CUYZ39 70681821 IC50 = 23.5 nM T93580 C9BP5R 70681822 IC50 = 28.7 nM T93580 CP6E4R 70681828 IC50 = 57.4 nM T93580 CBHO57 70681829 IC50 = 5.4 nM T93580 COQC31 70681830 IC50 = 17.4 nM T93580 CUF80Q 70681831 IC50 = 34.2 nM T93580 CXU67P 70681832 IC50 = 53.6 nM T93580 C45NUH 70681833 IC50 = 26.3 nM T93580 CV91MS 70681834 IC50 = 29.1 nM T93580 CDN0C4 70683924 IC50 = 12.9 nM T93580 CH2PL3 70683932 IC50 = 14.5 nM T93580 C8E4JH 70683933 IC50 = 14 nM T93580 CA27DC 70683934 IC50 = 38.6 nM T93580 CUC9K6 70686055 IC50 = 35.7 nM T93580 C48CLJ 70686056 IC50 = 23.9 nM T93580 C59QXF 70688191 IC50 = 38.2 nM T93580 C3S9IJ 70688192 IC50 = 8.6 nM T93580 C1S3IH 70690203 IC50 = 10.9 nM T93580 CJ5PK6 70690208 IC50 = 27.8 nM T93580 CL0JW1 70692374 IC50 = 79.3 nM T93580 CNW8O1 70692382 IC50 = 88.9 nM T93580 CM2KW1 70692383 IC50 = 18.9 nM T93580 C04XZL 70694433 IC50 = 16.3 nM T93580 CD5O8R 70694437 IC50 = 19.7 nM T93580 CTLH58 70696507 IC50 = 32.5 nM T93580 C3TV8N 70696508 IC50 = 22.3 nM T93580 D05AMQ 6539137 IC50 = 14.4 nM T93580 D0M5DR 57330144 IC50 = 54.3 nM T11764 D00STL 644241 IC50 < 2.54 nM T11764 D0AZ3C 5291 IC50 = 141 nM T11764 D0E6XR 3062316 IC50 = 0.4 nM T11764 D0P8IV 457193 IC50 = 9000 nM T11764 D0W5HK 216239 IC50 = 7 nM T11764 D00YPR 9811611 IC50 = 450 nM T11764 D02XNW 5494449 IC50 = 18 nM T11764 D0E3TC 44259 IC50 = 1.19 nM T11764 D03BNU 59604787 IC50 > 10000 nM T11764 D0D5PL 71577234 IC50 = 145 nM T11764 D0T3ME 156422 IC50 = 10 nM T11764 CP94XG 248316 IC50 = 80800 nM T11764 CIV15Q 10113978 IC50 = 51 nM T11764 C7E0YH 10896702 IC50 = 8 nM T11764 C5KNF9 10915062 IC50 = 2500 nM T11764 CS0G7J 23646852 IC50 = 408 nM T11764 CJ0CU5 24825841 IC50 = 3.1 nM T11764 C4FZ8E 24875320 IC50 = 18.6 nM T11764 C3DI7Y 24995523 IC50 = 82 nM T11764 CTO24B 25174101 IC50 = 487 nM T11764 C41MJN 25210518 IC50 = 558 nM T11764 CC6HK7 25210519 IC50 = 332 nM T11764 CFU8G9 25210521 IC50 = 856 nM T11764 CFK1A5 44473625 IC50 = 183 nM T11764 C61DVY 50990961 IC50 = 2.6 nM T11764 CV3UP9 50992247 IC50 = 7 nM T11764 CQR68T 50997019 IC50 = 5.5 nM T11764 C09ZRW 51035417 IC50 = 1150 nM T11764 C4PXI2 51035418 IC50 = 670 nM T11764 C2VAX9 51035420 IC50 = 19 nM T11764 CNWQ30 51035421 IC50 = 9170 nM T11764 C8NA4L 53384644 IC50 = 7000 nM T11764 C6N5LO 57328555 IC50 = 230 nM T11764 C9YFQ6 57328626 IC50 = 1670 nM T11764 CRX5L6 57328627 IC50 = 380 nM T11764 C6MW3N 57328628 IC50 = 1840 nM T11764 CC42AT 57839288 IC50 = 20 nM T11764 C5FN6H 57839380 IC50 = 30 nM T11764 CH7L5N 58172700 IC50 = 17.22 nM T11764 C2HN0Y 59553096 IC50 = 10900 nM T11764 C7SGT6 60202316 IC50 = 1 nM T11764 CV63UL 67240318 IC50 > 10000 nM T11764 CRH2Y9 68639605 IC50 = 100.56 nM T11764 CG1C2Y 70701953 IC50 = 76 nM T11764 C6HF8S 71521082 IC50 = 653.3 nM T11764 C9Z3AI 71521083 IC50 = 178.6 nM T11764 C1IT5U 71550931 IC50 = 101.4 nM T11764 CG1I5B 71550932 IC50 = 93.65 nM T11764 C1F5NV 71624671 IC50 > 1000 nM T11764 CQE01I 71624672 IC50 > 1000 nM T11764 CV8XI0 71624673 IC50 > 1000 nM T11764 CY82NR 71624674 IC50 > 1000 nM T11764 C0IM7Z 71624675 IC50 > 1000 nM T11764 C6JS8P 71624676 IC50 > 1000 nM T11764 C2F0QN 71624677 IC50 > 1000 nM T11764 CQ75IY 71624788 IC50 > 1000 nM T11764 C6GT1Q 71624789 IC50 > 1000 nM T11764 C6ZYR9 71624790 IC50 > 1000 nM T11764 CCSI30 71624792 IC50 > 1000 nM T11764 C4JD7I 71624793 IC50 > 1000 nM T11764 CS0AQ6 71624904 IC50 > 1000 nM T11764 C23XIU 71624905 IC50 > 1000 nM T11764 C4KTH9 71624906 IC50 > 1000 nM T11764 C7BG9F 71624907 IC50 > 1000 nM T11764 CC61DF 71624908 IC50 = 73.84 nM T11764 CRLN56 71624909 IC50 > 1000 nM T11764 CLO8V2 71625035 IC50 > 1000 nM T11764 CQI0N1 71625036 IC50 > 1000 nM T11764 CO41GB 71625037 IC50 > 1000 nM T11764 CC68IJ 71625038 IC50 = 2270 nM T11764 C4SV3X 71625039 IC50 > 1000 nM T11764 CT2K6M 71625040 IC50 = 116 nM T11764 C6JZ2E 71625161 IC50 > 1000 nM T11764 CRGQ64 71625290 IC50 = 37.1 nM T11764 CP83JY 71625291 IC50 = 103 nM T11764 CGJ8H4 71625292 IC50 = 125 nM T11764 C0D4LN 71625406 IC50 = 775.9 nM T11764 C9B1RV 71625407 IC50 = 214 nM T11764 CKOL80 71625408 IC50 = 131.36 nM T11764 CQY4U2 71625409 IC50 = 172.65 nM T11764 C42VJY 71764060 IC50 = 2 nM T11764 C6R8DI 72943374 IC50 = 64 nM T11764 CGDB30 74538658 IC50 = 290 nM T11764 CNR39Z 86763813 IC50 = 6.1 nM T11764 C9IZF3 86763814 IC50 = 1300 nM T11764 CR9V4A 86763924 IC50 = 8.1 nM T11764 CX94SV 86764031 IC50 = 4.5 nM T11764 C27YNT 86764144 IC50 = 5.8 nM T11764 CXW8T3 86764574 IC50 = 8.2 nM T11764 CTKA08 86764579 IC50 = 3.3 nM T11764 CI4HR3 90044151 IC50 = 15 nM T11764 CG46TN 90044499 IC50 = 6 nM T11764 COX57I 90656527 IC50 = 14400 nM T11764 C7FRI5 90656528 IC50 = 687 nM T11764 CQCX41 118737057 IC50 = 128 nM T11764 CN4X0C 121231414 IC50 = 188 nM T11764 C49UGP 122187122 IC50 = 280 nM T11764 CQL0W7 122197565 IC50 = 1400 nM T11764 CN41IF 122634050 IC50 = 457 nM T11764 CBYC49 126617676 IC50 = 349.6 nM T11764 C6RPF1 130364436 IC50 = 10000 nM T11764 CSY34O 130364443 IC50 = 6700 nM T11764 CI9H2W 130364450 IC50 = 514 nM T11764 CM4TO5 130364451 IC50 = 1800 nM T11764 CV4DH7 130364460 IC50 = 1500 nM T11764 CW91ZV 130364461 IC50 = 4500 nM T11764 CQIZ43 130364463 IC50 = 1100 nM T11764 C4IKC6 130364464 IC50 = 462 nM T11764 C0X6JS 130364465 IC50 = 846 nM T11764 C0ZGC1 130364467 IC50 = 944 nM T11764 CO9C5Q 130364468 IC50 = 8000 nM T11764 CQW3P1 130364471 IC50 = 1400 nM T11764 CHWX05 130364473 IC50 = 682 nM T11764 CLB65Y 130364478 IC50 = 940 nM T11764 CUZG19 130364481 IC50 > 10000 nM T11764 C34OMJ 130364482 IC50 = 3700 nM T11764 C6TWR3 130364484 IC50 = 2100 nM T11764 C8SF5Q 130364488 IC50 = 354 nM T11764 CS5C4E 130364494 IC50 = 2600 nM T11764 CVQ32Y 130364503 IC50 = 604 nM T11764 CV8B0Y 130364506 IC50 = 7600 nM T11764 CHX23J 130364524 IC50 = 1400 nM T11764 CHYL89 130364535 IC50 = 2200 nM T11764 C6OMB1 132204257 IC50 = 61 nM T11764 C6ROQ3 132546210 IC50 = 325 nM T11764 CQR94G 134198433 IC50 = 4500 nM T11764 C1X6FJ 134693894 IC50 = 20.4 nM T11764 CXC69T 137321158 IC50 = 116 nM T11764 CWC49K 137321210 IC50 = 21.5 nM T11764 C5VE4K 137636547 IC50 = 2600 nM T11764 C06JRX 137637094 IC50 = 0.8 nM T11764 CZ05TY 137637593 IC50 > 10000 nM T11764 CU9YQ3 137637635 IC50 > 10000 nM T11764 C6PKY7 137645383 IC50 > 10000 nM T11764 CHR9E0 137651685 IC50 = 203 nM T11764 CY53VO 137651787 IC50 > 10000 nM T11764 CE8DW7 137658399 IC50 > 10000 nM T11764 CU61WM 137658936 IC50 > 10000 nM T11764 CY9N8Q 137662234 IC50 = 255 nM T11764 CFR0X3 138454761 IC50 = 3.2 nM T11764 CM3A8O 139030333 IC50 = 5600 nM T11764 CB69CL 145925694 IC50 = 7.39 nM T11764 C7SH9V 145949579 IC50 = 7 nM T11764 CQCV54 145950906 IC50 = 1540 nM T11764 CKWZ34 145950923 IC50 = 10.4 nM T11764 CGOE73 145951398 IC50 = 47.4 nM T11764 CZF70O 145951916 IC50 = 83.1 nM T11764 CNK12Z 145952731 IC50 = 61.1 nM T11764 CW3RV1 145953992 IC50 > 10000 nM T11764 CGV16H 145954003 IC50 = 2100 nM T11764 CUIT87 145955254 IC50 = 34.1 nM T11764 CX2U6N 145956375 IC50 = 94.2 nM T11764 CC0RU9 145956925 IC50 = 4800 nM T11764 CA2F0O 145958559 IC50 = 13.1 nM T11764 C12VOP 145959821 IC50 = 2200 nM T11764 C5PZ9J 145959874 IC50 = 221 nM T11764 CF0C6K 145960274 IC50 = 45.3 nM T11764 CJDG56 145960632 IC50 > 10000 nM T11764 CE21QP 145961382 IC50 > 10000 nM T11764 CI0V8W 145963248 IC50 > 10000 nM T11764 C8NDS6 145971939 IC50 = 40.2 nM T11764 CP9NB6 145974090 IC50 = 3800 nM T11764 CI85EU 145998085 IC50 = 933 nM T11764 CD49VM 155295006 IC50 = 1740 nM T11764 CSHC63 155510467 IC50 = 196.7 nM T11764 CS0Y1T 155512636 IC50 = 3.8 nM T11764 CG09WO 155512858 IC50 > 5000 nM T11764 C6H8ZU 155513172 IC50 = 725 nM T11764 C2MD1Q 155513187 IC50 > 10000 nM T11764 CZDH58 155514096 IC50 > 5000 nM T11764 CDU75B 155514157 IC50 = 4.79 nM T11764 C79SJT 155514996 IC50 = 9.5 nM T11764 CB5T9G 155515436 IC50 = 207.3 nM T11764 CHAG14 155516692 IC50 = 1.2 nM T11764 CUHZ87 155516883 IC50 > 1000 nM T11764 C84GJO 155517474 IC50 = 1080 nM T11764 C9QXL4 155518155 IC50 = 8 nM T11764 C63PZX 155518871 IC50 = 3227 nM T11764 C1QO2I 155519342 IC50 = 1.5 nM T11764 CT0V6H 155519724 IC50 = 10.6 nM T11764 C7FIU3 155520706 IC50 = 3.2 nM T11764 C1ID9A 155523715 IC50 = 21.6 nM T11764 C1DY8F 155524432 IC50 = 6.5 nM T11764 CS1U2Z 155526433 IC50 = 3.7 nM T11764 CHD8E5 155527081 IC50 = 6.2 nM T11764 CFUG34 155527917 IC50 = 2.7 nM T11764 CNP8T7 155530083 IC50 = 135 nM T11764 CK10UA 155531677 IC50 = 1018 nM T11764 CS69CA 155532132 IC50 = 2.6 nM T11764 CFB02G 155532218 IC50 = 6.2 nM T11764 CURO30 155532620 IC50 = 6.36 nM T11764 CFY14G 155533271 IC50 = 6.7 nM T11764 C3PWI1 155534046 IC50 > 1000 nM T11764 CWLZ25 155535008 IC50 > 10000 nM T11764 CTXK93 155535665 IC50 = 102.2 nM T11764 C14SEB 155535950 IC50 = 634 nM T11764 C0ZP6C 155536159 IC50 = 67.9 nM T11764 C8NA6L 155536370 IC50 = 66.1 nM T11764 C91EQO 155536679 IC50 = 75.9 nM T11764 C3LC9I 155536820 IC50 = 3162.28 nM T11764 C65IAY 155537364 IC50 = 64.3 nM T11764 CI26FR 155538679 IC50 = 4.4 nM T11764 C3O6WX 155540330 IC50 > 1000 nM T11764 CXG71B 155540768 IC50 = 44.1 nM T11764 C3Q9UA 155541932 IC50 > 10000 nM T11764 C4G3ZT 155542710 IC50 = 3.9 nM T11764 CM96DX 155543017 IC50 = 2.7 nM T11764 C76NKG 155543431 IC50 > 1000 nM T11764 CC9LQ2 155546287 IC50 = 220 nM T11764 CI27QV 155546853 IC50 > 10000 nM T11764 CW4FU3 155546952 IC50 = 55.6 nM T11764 C5SXH4 155547874 IC50 = 2.6 nM T11764 CYP2O5 155547984 IC50 = 610 nM T11764 CD8A5R 155549158 IC50 = 8.8 nM T11764 CK86HR 155549476 IC50 = 3.4 nM T11764 C9MJL5 155551408 IC50 = 467 nM T11764 CX1L7G 155552114 IC50 = 4.7 nM T11764 CL8KR2 155552517 IC50 > 10000 nM T11764 CA9Y3J 155552522 IC50 = 4.56 nM T11764 C1TA9J 155553503 IC50 > 5000 nM T11764 C8BAU3 155554243 IC50 > 10000 nM T11764 CCQF25 155555943 IC50 = 1728 nM T11764 CFC8B0 155557936 IC50 = 2.6 nM T11764 CZ1TL4 155560174 IC50 = 7 nM T11764 CYD1C7 155560599 IC50 > 1000 nM T11764 C2EDK1 155562180 IC50 = 11 nM T11764 CHLY93 155562871 IC50 = 1326 nM T11764 CBG9Z1 155562952 IC50 > 1000 nM T11764 C2L5MS 155563171 IC50 = 2.9 nM T11764 C0WZ9S 155563842 IC50 > 1000 nM T11764 C60KLJ 155564326 IC50 > 10000 nM T11764 CAU45D 155565428 IC50 = 5.2 nM T11764 C4BS6J 155565938 IC50 = 947 nM T11764 CINX89 155566065 IC50 > 10000 nM T11764 C7Q4RY 155566792 IC50 = 663.5 nM T11764 C0V7SM 155567015 IC50 > 1000 nM T11764 C3MK6Z 155567552 IC50 = 8.7 nM T11764 CP69SU 155567937 IC50 = 2631 nM T11764 CF1W4I 155568065 IC50 = 7.7 nM T11764 D0BL0O 71624791 IC50 > 1000 nM T11764 D0N4LR 53469448 IC50 = 524 nM T11011 D0LI1C 44469321 IC50 > 30000 nM T11011 D0ZM5O 9884366 IC50 > 1000 nM T11011 CO9VA3 9820671 IC50 > 1000 nM T11011 C10HTZ 9869432 EC50 = 42 nM T11011 CA8CX9 9886113 Ki > 10000 nM T11011 C7SMT0 9908904 IC50 > 1000 nM T11011 C8LC4X 10112776 IC50 > 10000 nM T11011 C03DPR 10432407 IC50 > 10000 nM T11011 CAM63X 42618195 IC50 > 1000 nM T11011 C8K4UF 42618197 IC50 > 1000 nM T11011 C4MV2L 44290322 Ki > 10000 nM T11011 C8TQ1J 44321641 EC50 = 0.32 nM T11011 C2ZP0L 56661338 IC50 = 0.62 nM T11011 CWB2V7 56668206 IC50 = 46 nM T11011 CP2VR4 56668215 IC50 = 10 nM T11011 CAJ06Z 56675099 IC50 = 69 nM T11011 C96JRX 57912459 IC50 > 10000 nM T11011 CIS4J2 60155541 Ki > 10000 nM T11011 CBG90L 73345508 IC50 = 1.9 nM T11011 CCVD49 73345509 IC50 = 1.1 nM T11011 CS8D3J 73346924 IC50 = 4.9 nM T11011 C86PER 73348542 IC50 = 5.5 nM T11011 C3I5TA 73348776 Ki = 1.26 nM T11011 C24WZC 73349901 IC50 = 0.42 nM T11011 C8UXB0 73350007 IC50 > 500 nM T11011 C1KJ7S 73350131 IC50 = 1.3 nM T11011 CZ9LY3 73350133 IC50 > 100 nM T11011 C61OBY 73351508 IC50 = 60 nM T11011 CDF4S9 73351515 IC50 = 5 nM T11011 CN3V9Y 73351613 IC50 = 17.8 nM T11011 C45OSY 73351614 IC50 = 0.92 nM T11011 CO1H4V 73351615 IC50 = 0.51 nM T11011 CZH5L2 73351616 IC50 = 0.61 nM T11011 CW12AB 73353094 IC50 = 0.57 nM T11011 C91IUQ 73353095 IC50 = 81 nM T11011 CV07PY 73353096 IC50 = 6.2 nM T11011 CG9U8K 73353098 IC50 = 0.72 nM T11011 C1OV4F 73354615 IC50 = 1.3 nM T11011 CLIJ68 73354788 Ki = 12.2 nM T11011 CV18GL 73356172 IC50 = 0.6 nM T11011 CL78JX 73356174 IC50 = 1.2 nM T11011 C3KVB1 73356175 IC50 > 100 nM T11011 CR13BY 145969226 IC50 > 10000 nM T11011 D06FIF 9862166 Ki > 10000 nM T99802 D05MQK 110635 IC50 = 33 nM T99802 D0C9SY 135400189 IC50 = 240 nM T99802 D0F9GE 3108 Ki = 400 nM T99802 D0Z7ZM 135398744 IC50 = 3000 nM T99802 D01LCC 17754438 IC50 > 10000 nM T99802 D0T5PO 5092 IC50 > 16000 nM T99802 D0X0PP 59351313 IC50 > 30000 nM T99802 D05VBJ 71295299 IC50 = 6920 nM T99802 D0WS3T 72706254 IC50 = 280 nM T99802 D00YPW 135399235 Ki = 12000 nM T99802 D01FXD 9802841 IC50 > 10000 nM T99802 C1B6ZL 662965 IC50 > 50000 nM T99802 C8JLO0 2243267 IC50 = 2300 nM T99802 CZH08Y 9802738 IC50 = 219 nM T99802 C3AOI5 10138533 IC50 = 53 nM T99802 CDJ0T8 10272508 IC50 = 73 nM T99802 C90QZM 10324834 IC50 = 5.5 nM T99802 C45VZC 11438405 IC50 = 11600 nM T99802 C4ZYH9 11547485 IC50 = 540 nM T99802 CX0FM3 11547713 IC50 = 2200 nM T99802 CHU90R 11598626 IC50 = 2300 nM T99802 C1G3EI 11620160 IC50 = 2200 nM T99802 C6GY9D 11635241 IC50 = 2100 nM T99802 CXD82O 11649109 IC50 = 2000 nM T99802 CA26IK 11742611 IC50 = 7300 nM T99802 CUK49V 11988837 Ki = 2600 nM T99802 CFIO49 11988967 Ki = 7100 nM T99802 C2D0NG 11989101 Ki = 28000 nM T99802 C65ABT 11989102 Ki = 72000 nM T99802 C1B4XD 11992634 IC50 = 64.1 nM T99802 CPX16N 11993169 IC50 = 346 nM T99802 COG39H 16727125 IC50 = 1000 nM T99802 CW96SI 23624262 IC50 = 68.6 nM T99802 CJ0ZF1 24180492 IC50 = 2000 nM T99802 C9WGI4 24802717 IC50 = 690 nM T99802 CC5MR8 24810057 IC50 = 7700 nM T99802 CO0QJ5 24810103 IC50 = 24300 nM T99802 C30GDM 24810105 IC50 = 9500 nM T99802 C1GV0Y 24810146 IC50 = 7800 nM T99802 CN27KS 24810195 IC50 = 10500 nM T99802 COI6Q5 24810296 IC50 = 5700 nM T99802 CLN9Q4 24810297 IC50 = 5200 nM T99802 C4H6WK 24810298 IC50 = 12000 nM T99802 CU1IL5 24810299 IC50 = 7700 nM T99802 CY4VE3 24810442 IC50 = 14700 nM T99802 C37QID 24810545 IC50 = 7100 nM T99802 CP8K1E 24810599 IC50 = 39300 nM T99802 CTX94M 24810757 IC50 = 22700 nM T99802 C20VHK 24871823 IC50 = 3030 nM T99802 CA9PN0 24957913 IC50 = 85 nM T99802 CICF39 42629702 IC50 > 10000 nM T99802 CM3X9S 42629827 IC50 > 1000 nM T99802 CQN26J 42629945 IC50 = 2400 nM T99802 C6O5FX 42630062 IC50 = 2810 nM T99802 C71ZNR 42630180 IC50 = 1510 nM T99802 C4RHY0 42630191 IC50 > 10000 nM T99802 CT6RS9 42630192 IC50 = 2200 nM T99802 CYZL43 42630317 IC50 = 4870 nM T99802 CH42OZ 42630318 IC50 = 3350 nM T99802 C7X5AH 42630437 IC50 = 2350 nM T99802 CW8OB3 44243146 Ki = 14600 nM T99802 CV1ZA7 44280486 IC50 = 4.3 nM T99802 CG8R0W 44280487 IC50 = 4.7 nM T99802 CS0FX4 44280546 IC50 = 6.7 nM T99802 C05SIA 44280556 IC50 = 6.5 nM T99802 CA9KV4 44280558 IC50 = 48 nM T99802 CY74KE 44280614 IC50 = 48 nM T99802 C4RO9D 44280635 IC50 = 4.7 nM T99802 CH7W2T 44280722 IC50 = 3.5 nM T99802 CTO54N 44280723 IC50 = 2.2 nM T99802 CXRU70 44280792 IC50 = 31 nM T99802 CO7NV0 44280794 IC50 = 950 nM T99802 CDQ8B2 44280847 IC50 = 2.01 nM T99802 C0N3JE 44280911 IC50 = 4.2 nM T99802 C3DHJ2 44280985 IC50 = 2.4 nM T99802 CA3GF6 44280994 IC50 = 39 nM T99802 CXB40D 44281036 IC50 = 11.8 nM T99802 CA1HN8 44281061 IC50 = 43 nM T99802 C7TKW4 44281095 IC50 = 22 nM T99802 CK3W1B 44281096 IC50 = 118 nM T99802 CC81DV 44281265 IC50 = 71 nM T99802 CNO94A 44281273 IC50 = 1000 nM T99802 C1NZE3 44441802 IC50 = 7600 nM T99802 CM13IX 44441825 IC50 = 820 nM T99802 CSD1Q8 44441827 IC50 = 600 nM T99802 CG49SA 44441829 IC50 = 500 nM T99802 C8FK0V 44441831 IC50 = 1500 nM T99802 CTI03C 44441833 IC50 = 130 nM T99802 CZYW49 44441837 IC50 = 970 nM T99802 CQ0N7Y 44441840 IC50 = 3300 nM T99802 CWB9V3 46226892 IC50 = 5000 nM T99802 C5IMB2 46239424 Ki = 1900 nM T99802 CKR9P7 46239425 Ki = 6600 nM T99802 C7SLP0 46239531 Ki = 1200 nM T99802 CI1F5C 46239840 Ki >= 770 nM T99802 C26XVS 46240044 Ki >= 4793 nM T99802 CE4JU7 46842025 IC50 > 10000 nM T99802 CR8JC2 46842169 IC50 > 10000 nM T99802 C3P2IN 46933992 IC50 >= 95000 nM T99802 CHA5Z0 49821469 IC50 > 1000 nM T99802 C1AYP0 49821627 IC50 > 500 nM T99802 C85AXR 49821714 IC50 > 1000 nM T99802 CZS03D 50902030 Ki > 4274 nM T99802 CH2Z1E 50902289 Ki > 7100 nM T99802 C4HJL2 50902291 Ki > 7950 nM T99802 C6A1IU 50902549 Ki > 2000 nM T99802 C3Y2AV 50903255 Ki > 2000 nM T99802 CN41YJ 50925469 IC50 = 104 nM T99802 CQ3RG5 50925470 IC50 = 1500 nM T99802 CBT56Y 54581676 IC50 = 140 nM T99802 CGF65A 54670110 IC50 > 30000 nM T99802 C90ZLC 54670399 IC50 > 30000 nM T99802 C4TGL7 56648496 IC50 > 1000 nM T99802 CH6C3L 56648679 IC50 > 10000 nM T99802 CCY79V 56648680 IC50 = 5090 nM T99802 CNE96P 56648857 IC50 = 5290 nM T99802 CX86AQ 56648859 IC50 > 5000 nM T99802 CPC3T4 56654131 IC50 > 10000 nM T99802 C0YD3P 56928304 IC50 > 5000 nM T99802 C8RO6A 56929788 IC50 > 1000 nM T99802 CG3DF1 57392948 Ki > 10000 nM T99802 CE36TV 57394695 Ki = 2300 nM T99802 CPA3D1 57403394 Ki = 4900 nM T99802 CDA74Z 57600658 IC50 = 2300 nM T99802 C6FY8M 57600737 IC50 = 1100 nM T99802 CR6Z9C 57600809 IC50 = 1800 nM T99802 C2PGE3 57600813 IC50 = 1600 nM T99802 CLK8O5 57600820 IC50 = 4800 nM T99802 C7O5HY 57600960 IC50 = 1400 nM T99802 CK7L8X 57601096 IC50 = 1100 nM T99802 CN8D4I 57601175 IC50 = 1300 nM T99802 C0PXR1 57601304 IC50 = 1400 nM T99802 CNH5Y7 57601312 IC50 = 3900 nM T99802 C81JFC 57601337 IC50 = 2500 nM T99802 C6LY3S 57601465 IC50 = 2100 nM T99802 CYM0K3 57601557 IC50 = 2700 nM T99802 C2IPY1 57601592 IC50 = 870 nM T99802 CVB98S 57601701 IC50 = 1100 nM T99802 CD5CJ9 57601760 IC50 = 2700 nM T99802 CL3EN6 57601817 IC50 = 2700 nM T99802 C1HF7E 57601851 IC50 = 3400 nM T99802 C57LTR 57602000 IC50 = 1100 nM T99802 C6XR8W 57602004 IC50 = 3600 nM T99802 C4XMB6 58547809 IC50 > 30000 nM T99802 CEB3G9 58547814 IC50 > 30000 nM T99802 C08QVG 58547833 IC50 > 30000 nM T99802 CFVG67 58547863 IC50 > 30000 nM T99802 CYZA38 58548077 IC50 = 10600 nM T99802 CWX3N7 59320301 IC50 = 963 nM T99802 C0EP5I 59341847 IC50 > 10000 nM T99802 CHQ28A 59341978 IC50 > 10000 nM T99802 CY8J3O 68181896 IC50 > 10000 nM T99802 CC43LF 71074083 IC50 > 10000 nM T99802 C4P0XT 71092344 IC50 > 30000 nM T99802 C6DAG4 71092519 IC50 > 30000 nM T99802 C2HGI7 71153408 IC50 = 2138 nM T99802 C9GR3L 71153436 IC50 > 10000 nM T99802 C4GNJ3 71598545 IC50 > 1000 nM T99802 C68SDB 71719394 IC50 = 1995.26 nM T99802 CZ0G2X 72165213 IC50 > 10000 nM T99802 C7XRY6 72190879 IC50 > 30000 nM T99802 CQ3GD7 72704434 Ki = 1300 nM T99802 CBM61I 73293715 IC50 = 2440 nM T99802 C9JE6M 75815419 IC50 = 34.7 nM T99802 CF03DW 90168772 IC50 > 20000 nM T99802 CM6J9K 90168778 IC50 > 20000 nM T99802 CSCY01 117949009 IC50 > 10000 nM T99802 CYQ74R 118479645 IC50 > 10000 nM T99802 CVYK24 118556943 IC50 > 20000 nM T99802 CRJE23 122185011 IC50 = 8257 nM T99802 CS6M9C 122193679 IC50 > 100000 nM T99802 C4UR7D 127038167 IC50 > 1000 nM T99802 C4H2TJ 127038168 IC50 > 1000 nM T99802 CL9JT8 127038169 IC50 = 494 nM T99802 CJPX60 127038509 IC50 = 286 nM T99802 C26EAG 127038511 IC50 > 1000 nM T99802 CTM9E4 127038512 IC50 = 286 nM T99802 C6AQ2U 127038513 IC50 = 413 nM T99802 CV1FM0 127038868 IC50 = 395 nM T99802 CADU23 127038869 IC50 = 457 nM T99802 CJ94GK 129316454 IC50 = 5060 nM T99802 C2P1IU 134129996 IC50 > 100000 nM T99802 C0A1CZ 134131162 IC50 > 100000 nM T99802 CHDC83 135566745 IC50 = 3360 nM T99802 C21FVA 136180322 IC50 = 1400 nM T99802 CQW7T0 136197286 IC50 = 998 nM T99802 C2N9VT 137348687 IC50 > 10000 nM T99802 CPTE92 138319693 IC50 = 39 nM T99802 C2QLX3 138393292 IC50 > 50000 nM T99802 CF3B2O 141492937 IC50 = 2.7 nM T99802 C93ZIQ 141492999 IC50 = 5.1 nM T99802 C0JV6Y 141737649 IC50 = 153 nM T99802 CSOF52 141737655 IC50 > 1000 nM T99802 C7SRA2 141737657 IC50 = 169 nM T99802 CMIY07 141737666 IC50 = 155 nM T99802 CC61SD 141737667 IC50 > 1000 nM T99802 C14CZJ 141737668 IC50 = 99 nM T99802 CTNG49 141737674 IC50 = 386 nM T99802 CJ38IC 141737676 IC50 = 119 nM T99802 C1MC5Z 141737681 IC50 = 173 nM T99802 CTUL23 141737690 IC50 > 1000 nM T99802 CMW20N 141737696 IC50 = 272 nM T99802 C7GBH6 141737698 IC50 = 634 nM T99802 CO1C4S 141737703 IC50 = 802 nM T99802 CX9N1P 141737704 IC50 = 4 nM T99802 C8HEG7 141737705 IC50 > 1000 nM T99802 C1S7HV 142592633 IC50 = 1500 nM T99802 CN3OC2 142592634 IC50 = 250 nM T99802 CY64NR 142592636 IC50 = 245 nM T99802 C83XNL 142592649 IC50 = 480 nM T99802 C7XZB1 142592652 IC50 = 659 nM T99802 CC7HN2 145974174 IC50 > 100000 nM T99802 CK1BR0 145978345 IC50 > 100000 nM T99802 CL8CU6 155521936 IC50 > 200000 nM T99802 CT85RG 155530589 IC50 > 200000 nM T99802 D06NIT 135564899 IC50 > 1000 nM T99802 D09RKU 46239428 Ki = 1600 nM T99802 D0V4WB 149790 IC50 > 16000 nM T68163 D00STL 644241 IC50 = 1281 nM T68163 D04LVK 57379345 IC50 = 840 nM T68163 D09KTS 24821094 IC50 = 200 nM T68163 D0AZ3C 5291 IC50 = 220 nM T68163 D0E6XR 3062316 IC50 = 1.2 nM T68163 D0H0EQ 24826799 IC50 = 0.24 nM T68163 D0J9ZR 4477 IC50 = 23800 nM T68163 D0OB0F 5328940 IC50 = 8 nM T68163 D02LJW 23635314 IC50 = 100 nM T68163 D02RJY 11442891 IC50 > 10000 nM T68163 D02UFQ 11620908 IC50 = 5200 nM T68163 D03HUX 49792852 IC50 > 10000 nM T68163 D03LWG 53235510 IC50 = 3019 nM T68163 D04BFC 59174488 IC50 = 4400 nM T68163 D07EHV 44814409 IC50 > 10000 nM T68163 D07HPJ 11476171 IC50 = 1400 nM T68163 D08UUL 46700756 IC50 > 10000 nM T68163 D0E3TC 44259 IC50 = 0.49 nM T68163 D0G0VV 11387605 IC50 = 11 nM T68163 D0H9FR 118295624 IC50 = 631 nM T68163 D0M9QZ 11485656 IC50 > 50000 nM T68163 D0Q9UX 16718576 IC50 > 10000 nM T68163 D0R9IU 44462758 IC50 = 238 nM T68163 D0S6TK 11213558 IC50 = 732 nM T68163 D0Z4RC 24756910 IC50 = 840 nM T68163 D03BNU 59604787 IC50 > 10000 nM T68163 D00OWF 5280953 IC50 > 250000 nM T68163 D0WX0K 71680628 IC50 = 170 nM T68163 D08DBE 10344820 Ki = 30 nM T68163 D09HEV 6539952 IC50 = 29 nM T68163 D0T3ME 156422 IC50 = 960 nM T68163 C1ZG2U 449087 IC50 > 10000 nM T68163 CUEZ35 5330437 IC50 = 140 nM T68163 CDK3J0 5703619 IC50 = 4 nM T68163 CPXK25 5793057 IC50 > 100000 nM T68163 CB7WK3 5938113 IC50 = 10500 nM T68163 CP0XI6 6603792 IC50 = 420 nM T68163 CY3MK1 9807952 IC50 = 8.5 nM T68163 CM5Z8X 9869943 IC50 = 2 nM T68163 C1W4JG 9872939 IC50 = 1000 nM T68163 C5GE7T 9917045 IC50 = 2400 nM T68163 C6RI8P 9986150 IC50 = 230 nM T68163 CLI9A3 10029363 IC50 = 35 nM T68163 CT9F2H 10053560 IC50 = 4.8 nM T68163 CINF40 10073694 IC50 = 1800 nM T68163 CSGD16 10246246 IC50 > 7000 nM T68163 CPS79C 10402283 IC50 < 10 ug.mL-1 T68163 C7TJ9U 10483163 IC50 = 3.1 nM T68163 CMQA73 11215316 IC50 = 3.4 nM T68163 CVOW82 11238420 IC50 = 5300 nM T68163 CBOP58 11293798 Ki > 10000 nM T68163 C26BZX 11362471 Ki > 10000 nM T68163 CB45PJ 11362483 IC50 = 275 nM T68163 C25ZCN 11374110 IC50 > 50000 nM T68163 CWXB93 11397177 Ki > 10000 nM T68163 CREQ51 11429654 IC50 > 50000 nM T68163 CY0A4E 11429729 IC50 > 50000 nM T68163 CFJ6B2 11441375 IC50 = 27 nM T68163 C4Q7XD 11474276 IC50 = 88 nM T68163 C8AY3B 11518031 IC50 < 25 nM T68163 C7HMO6 11526786 IC50 > 30000 nM T68163 CTG83F 11539329 Ki > 1700 nM T68163 CACS26 11561968 Ki > 2000 nM T68163 CMIL86 11590363 Ki > 1700 nM T68163 C69FYK 11604142 Ki = 400 nM T68163 C9T6SC 11640926 Ki > 1700 nM T68163 CJ9KN7 11683817 IC50 > 10000 nM T68163 CU0E8O 11690457 Ki > 2000 nM T68163 CB0AP2 11705863 Ki > 10000 nM T68163 CZY05V 11719421 IC50 = 21 nM T68163 C45EWD 11723489 IC50 > 7000 nM T68163 CE0KI4 11753519 IC50 = 12900 nM T68163 CP7AH3 11755812 IC50 = 6000 nM T68163 C9JT4S 11847343 IC50 > 10000 nM T68163 C5CPV2 12516472 IC50 = 10 ug.mL-1 T68163 C0M7TW 15948947 IC50 = 28 nM T68163 C1VNB4 15948949 IC50 = 5 nM T68163 CH8ZG5 15949048 IC50 = 9 nM T68163 CK2Z6Y 15949521 IC50 = 82 nM T68163 CBZF29 15949522 IC50 = 133 nM T68163 C34MCY 15949523 IC50 = 6 nM T68163 CS3P9G 15949524 IC50 = 10 nM T68163 C1KPH2 15949525 IC50 = 3296 nM T68163 C5JG9R 15949617 IC50 = 5 nM T68163 C8FT6U 15949618 IC50 = 332 nM T68163 C30PVQ 15949619 IC50 = 96 nM T68163 C3PNO2 15949620 IC50 = 88 nM T68163 C4I5RS 15949621 IC50 > 10000 nM T68163 CVJ9A0 15949712 IC50 = 30 nM T68163 CEI2K8 15949887 IC50 = 215 nM T68163 CAIN63 15949888 IC50 > 10000 nM T68163 C2VDI1 15949889 IC50 = 400 nM T68163 COC02T 15949890 IC50 = 1422 nM T68163 CFQ6X3 15949974 IC50 = 204 nM T68163 CMKZ23 15949975 IC50 = 642 nM T68163 CWM5L4 15949976 IC50 = 149 nM T68163 CO7NG2 15950141 IC50 = 217 nM T68163 COIG45 15950224 IC50 = 14 nM T68163 C9V0TO 15950311 IC50 = 15 nM T68163 CFPW41 16007116 Ki > 1600 nM T68163 C09OWB 16015442 IC50 = 500 nM T68163 C9TU1O 16046126 IC50 > 1000 nM T68163 CQG45C 16109001 IC50 = 4900 nM T68163 C1U8XW 16109036 IC50 = 180 nM T68163 CGC34R 16118737 IC50 = 0.9 nM T68163 CR92JO 16124248 IC50 = 37000 nM T68163 CP2M4O 16124345 IC50 = 100 nM T68163 C6TQ2O 16664354 Ki = 4.19 nM T68163 CDZ31W 16747696 IC50 > 50000 nM T68163 CWH37T 17758574 IC50 > 30000 nM T68163 CJA0D6 18451024 IC50 = 3700 nM T68163 C6FQB7 18451036 IC50 = 1180 nM T68163 C6JV7W 23400934 IC50 > 7000 nM T68163 CD5S7O 23401001 IC50 > 7000 nM T68163 CE7K3W 23532567 IC50 > 10000 nM T68163 CW6OB1 23627212 IC50 = 730 nM T68163 CK5N6B 23657635 IC50 = 40 nM T68163 CA3I4T 24753787 IC50 > 50000 nM T68163 CQNP54 24764449 IC50 = 506 nM T68163 C2UOE0 24766030 IC50 = 28 nM T68163 CJUK39 24770517 IC50 > 10000 nM T68163 C9PA0M 24807809 IC50 > 30000 nM T68163 CY8X0J 24811794 Ki > 10000 nM T68163 C9F1AO 24821023 IC50 = 200 nM T68163 CM28WD 24825721 IC50 > 10000 nM T68163 C1SVT2 24854903 IC50 = 954 nM T68163 CSW5V3 24865437 IC50 > 100000 nM T68163 C4V9GI 24960018 IC50 = 17000 nM T68163 CD5HQ0 24969301 IC50 > 10000 nM T68163 CS3Q8B 24995659 IC50 > 2000 nM T68163 C0B7RT 25057409 IC50 > 10000 nM T68163 C6P1CX 25066843 IC50 = 520 nM T68163 CSNC57 25110758 IC50 > 10000 nM T68163 C0GOX5 25110759 IC50 > 10000 nM T68163 CC2R7S 25110760 IC50 > 10000 nM T68163 CL82CU 25110796 IC50 > 1000000 nM T68163 C36FXD 25138012 IC50 = 3 nM T68163 CP6N4G 25138050 IC50 = 430 nM T68163 C57PDK 25191024 IC50 > 1000000 nM T68163 CR0S2O 25195244 IC50 = 23 nM T68163 CTX60V 25195245 IC50 = 74 nM T68163 CRO09K 25211064 IC50 = 58 nM T68163 C8B6TY 42628503 EC50 < 500 nM T68163 CLW80F 44160269 IC50 = 19000 nM T68163 CK73NR 44219749 IC50 > 50000 nM T68163 CEL61X 44229839 IC50 = 3000 nM T68163 CIX8V2 44251637 IC50 = 30000 nM T68163 CG1C9E 44269392 IC50 > 250000 nM T68163 CAT6W7 44269404 IC50 > 250000 nM T68163 C4SA3Y 44269518 IC50 > 250000 nM T68163 CO81DL 44318069 IC50 = 20 ug.mL-1 T68163 CEX4Q9 44430662 IC50 = 7.6 nM T68163 CYB28E 44430665 IC50 = 29 nM T68163 CA98KR 44432441 IC50 > 10000 nM T68163 CGV37F 44440254 IC50 = 20806 nM T68163 C5JUV3 44440256 IC50 > 50000 nM T68163 CFB56S 44440259 IC50 = 30587 nM T68163 CEW9G2 44440261 IC50 > 50000 nM T68163 CHZ8Y2 44449452 IC50 = 3400 nM T68163 C9Z8XJ 44460238 IC50 > 20 ug.mL-1 T68163 CV1Q0D 44460258 IC50 = 20 ug.mL-1 T68163 C5WL1F 44473009 IC50 = 5100 nM T68163 CEG1S5 44473011 IC50 = 9600 nM T68163 C46OMR 44473016 IC50 = 20000 nM T68163 C4WRN5 44541014 IC50 = 27.7 nM T68163 C3VRO9 44557921 IC50 > 10000 nM T68163 C8X1JW 44570801 IC50 = 410 nM T68163 CD9BY2 44570802 IC50 = 2200 nM T68163 C5BNG9 44570803 IC50 = 310 nM T68163 CC58RY 44570848 IC50 = 230 nM T68163 CGWK29 44570849 IC50 = 1700 nM T68163 CJY8S0 44570884 IC50 = 13000 nM T68163 C9VXN3 44578709 IC50 = 4000 nM T68163 C6FJ7Y 44589021 IC50 > 1000000 nM T68163 C28QLM 44605035 IC50 > 50000 nM T68163 C75XHS 44605037 IC50 > 50000 nM T68163 CU3RF1 45139989 IC50 > 10000 nM T68163 CQGZ06 45139991 IC50 > 10000 nM T68163 C2JVA4 45270368 IC50 = 40 nM T68163 CC95PQ 45375865 IC50 = 290 nM T68163 CEOQ27 45375866 IC50 > 50000 nM T68163 C5S8MA 45485083 IC50 = 520 nM T68163 CW42YX 45487634 IC50 > 5000 nM T68163 C96BNW 46179972 IC50 = 7 nM T68163 CZBL95 46220496 IC50 = 140 nM T68163 CY3HW5 46224684 IC50 > 10000 nM T68163 C7ON5A 46233287 IC50 > 10000 nM T68163 CQW97N 46846072 IC50 = 540 nM T68163 C7H4YM 46865419 IC50 > 10000 nM T68163 CC2O9R 46865656 IC50 = 3981.07 nM T68163 CO3P0J 46866604 IC50 < 50000 nM T68163 CLS29B 46872626 IC50 > 10000 nM T68163 CRS61F 46879438 IC50 > 10000 nM T68163 C27JEF 46879439 IC50 = 1384 nM T68163 CF0T8P 46879440 IC50 = 1315 nM T68163 C12RMW 46879441 IC50 = 1658 nM T68163 CH2D7N 46879442 IC50 = 1228 nM T68163 CI6OD8 46879443 IC50 = 134 nM T68163 C7YD4Q 46879444 IC50 = 113 nM T68163 C8MN5Q 46879445 IC50 = 84 nM T68163 CX6SW2 46879446 IC50 = 468 nM T68163 CNF3V6 46879447 IC50 = 8012 nM T68163 CW46VY 46879448 IC50 = 43 nM T68163 CLK6X3 46879907 IC50 = 3608 nM T68163 CRPU47 46879908 IC50 = 7 nM T68163 C1TIE9 46880013 IC50 = 595 nM T68163 C2A8KO 46880066 IC50 = 1471 nM T68163 CBRP80 46880067 IC50 = 1117 nM T68163 C3FY2B 46880068 IC50 = 457 nM T68163 CX89TY 46880069 IC50 = 399 nM T68163 CB0XY1 46880070 IC50 = 67 nM T68163 CUD81V 46880071 IC50 = 818 nM T68163 CZP58Q 46880072 IC50 = 547 nM T68163 CC8OF9 46880073 IC50 = 259 nM T68163 CF41HG 46880098 IC50 = 126 nM T68163 C6O2YG 46880099 IC50 = 1079 nM T68163 CI78DM 46880100 IC50 = 15 nM T68163 CU04ZK 46880101 IC50 = 16 nM T68163 C4E0MF 46880133 IC50 = 100 nM T68163 COJ16A 46880134 IC50 = 272 nM T68163 C71MGJ 46880135 IC50 > 10000 nM T68163 CJOM49 46880136 IC50 = 1760 nM T68163 C3R6TL 46880213 IC50 = 437 nM T68163 CT8BQ4 46880214 IC50 = 5512 nM T68163 C0JTO4 46880215 IC50 = 7836 nM T68163 CAFN49 46880216 IC50 > 10000 nM T68163 CRE96X 46885625 IC50 = 398 nM T68163 C2O8RZ 46886323 IC50 = 26 nM T68163 C9PAT7 46927672 IC50 = 10 nM T68163 CHSF07 49806372 IC50 > 1000 nM T68163 CF91RS 49843531 IC50 > 10000 nM T68163 C2Y6QS 50938552 IC50 > 10000 nM T68163 C9NYP4 51036677 IC50 > 10000 nM T68163 C4WRY3 51037112 IC50 > 10000 nM T68163 CRI28Z 51037948 IC50 > 10000 nM T68163 CEQN27 52936621 Ki > 1000 nM T68163 CD4H3S 53354074 Ki > 1000 nM T68163 C8NA4L 53384644 IC50 = 43000 nM T68163 CJBL48 56925034 IC50 = 68 nM T68163 C87YOZ 56929808 IC50 = 170 nM T68163 CR16SD 56947170 IC50 = 1360 nM T68163 CI6QE5 56970263 IC50 < 500 nM T68163 CPHX64 57325478 IC50 > 50000 nM T68163 CQ9BW4 57325479 IC50 > 50000 nM T68163 CQGH97 57391046 IC50 = 1670 nM T68163 C8GQ9H 57391143 IC50 = 10.9 nM T68163 CSU96R 57391144 IC50 = 490 nM T68163 C7OQ2B 57391145 IC50 = 7400 nM T68163 C3X1ZN 57392910 IC50 = 1420 nM T68163 COC5U3 57392911 IC50 = 327 nM T68163 CN03CZ 57392994 IC50 = 10.9 nM T68163 C2DRH3 57392995 IC50 = 533 nM T68163 CE1A9V 57394653 IC50 = 353 nM T68163 CIQH60 57394654 IC50 = 3080 nM T68163 CD5Z9R 57394655 IC50 = 1300 nM T68163 CNV76Z 57394656 IC50 = 3020 nM T68163 CO34BP 57394657 IC50 = 19 nM T68163 CH2PZ8 57396405 IC50 = 3730 nM T68163 CN8I2E 57396406 IC50 = 560 nM T68163 C3NG0U 57396491 IC50 = 46.6 nM T68163 CNC84H 57396492 IC50 = 1980 nM T68163 COG41M 57398104 IC50 = 378 nM T68163 C83EBV 57398105 IC50 = 2320 nM T68163 CL78SU 57398205 IC50 = 350 nM T68163 CVRX72 57398206 IC50 = 1590 nM T68163 C05PSA 57398207 IC50 = 40 nM T68163 CBK0C1 57399762 IC50 = 44.4 nM T68163 C4CQR0 57399857 IC50 = 6020 nM T68163 COC32E 57401532 IC50 = 167 nM T68163 C7Z4PU 57401624 IC50 = 1.55 nM T68163 C7M2NU 57401629 IC50 = 2130 nM T68163 CET8G9 57401630 IC50 = 3450 nM T68163 C1CJ3Y 57401631 IC50 = 2000 nM T68163 CCT87N 57401632 IC50 = 10400 nM T68163 CDS7G4 57401633 IC50 = 130 nM T68163 C5THG9 57401721 IC50 = 297 nM T68163 C6LWX8 57401722 IC50 = 623 nM T68163 CU1C9S 57401723 IC50 > 50000 nM T68163 CZ4UR3 57403361 IC50 = 716 nM T68163 CY1Z7M 57403363 IC50 = 19600 nM T68163 CG0Y3M 57403447 IC50 = 21.3 nM T68163 CVK0G4 58056356 IC50 > 50000 nM T68163 CH7L5N 58172700 IC50 = 3534 nM T68163 CZ3TG1 59375154 IC50 = 204 nM T68163 C1MR8Q 60097495 IC50 > 10000 nM T68163 CE49GC 67098566 Ki = 490 nM T68163 CV63UL 67240318 IC50 > 10000 nM T68163 C8I7GC 68293638 IC50 = 9800 nM T68163 CAIO65 68796885 IC50 = 37 nM T68163 C7VJ6A 70647728 IC50 = 160 nM T68163 C6U2WZ 70687578 IC50 = 352 nM T68163 C1IEJ2 70789254 IC50 = 178000 nM T68163 C8T7ZP 70789255 IC50 = 14000 nM T68163 COU73Y 71226944 IC50 = 74 nM T68163 C40JOZ 71235465 IC50 = 268 nM T68163 CEBO91 71452977 IC50 = 3300 nM T68163 CKT60L 71455860 Ki > 1600 nM T68163 C6HF8S 71521082 IC50 = 45420 nM T68163 C9Z3AI 71521083 IC50 = 15150 nM T68163 CCN01X 71547862 IC50 > 10000 nM T68163 CZ31PU 71583657 IC50 = 3000 nM T68163 CZM1K4 71765510 IC50 = 54 nM T68163 CZ97VP 86294733 IC50 = 1195 nM T68163 CPG3A5 86302574 IC50 > 30000 nM T68163 CY0UC4 90645194 IC50 > 10000 nM T68163 CV9H8U 90656285 IC50 = 190 nM T68163 CG7E1U 90656286 IC50 = 1800 nM T68163 CDF9O2 90656287 IC50 = 550 nM T68163 CY7BI2 118706214 IC50 > 10000 nM T68163 CDSV38 121316062 Ki = 190 nM T68163 C08KEM 122179540 IC50 = 7500 nM T68163 C3AJ4C 122179546 IC50 = 6400 nM T68163 CG0RP7 122179547 IC50 = 3400 nM T68163 C1A0SQ 122179548 IC50 = 4900 nM T68163 C5B6QT 122189918 IC50 = 65.9 nM T68163 CFKD32 122191637 IC50 = 824 nM T68163 C4X7SD 122192466 IC50 > 10000 nM T68163 C8F0DQ 129909860 IC50 = 31 nM T68163 CHS5X0 135409466 IC50 = 5 ug.mL-1 T68163 C2DH1R 135412832 IC50 = 18 ug.mL-1 T68163 CI47VJ 135566923 IC50 = 112 nM T68163 CZFA70 135611366 IC50 = 1255 nM T68163 CX4ZB3 135863110 IC50 = 8500 nM T68163 C5XIE8 136026041 IC50 = 14000 nM T68163 CO0L9T 136056541 IC50 = 44 nM T68163 CLIE18 136056542 IC50 = 1003 nM T68163 CM7V8J 136056543 IC50 > 10000 nM T68163 C64BEV 136056544 IC50 = 32 nM T68163 CP1MX4 136056545 IC50 = 230 nM T68163 C4AR8N 136056546 IC50 = 84 nM T68163 CC10GD 136056547 IC50 = 315 nM T68163 CN1PY3 136056548 IC50 = 69 nM T68163 CI8Y0U 136056549 IC50 > 10000 nM T68163 CVIC49 136069671 IC50 = 1400 nM T68163 C2U0DL 136185991 IC50 >> 5 ug.mL-1 T68163 CD48LY 136185992 IC50 = 5 ug.mL-1 T68163 CPE2B1 136185998 IC50 = 10 ug.mL-1 T68163 CR9XE0 136185999 IC50 > 20 ug.mL-1 T68163 C1I8LC 136186000 IC50 > 20 ug.mL-1 T68163 C40HWO 136186001 IC50 = 20 ug.mL-1 T68163 CGP04W 136186009 IC50 > 20 ug.mL-1 T68163 CS5QE7 136186010 IC50 > 20 ug.mL-1 T68163 CXC69T 137321158 IC50 = 85 nM T68163 CZOD53 137633880 IC50 = 646 nM T68163 C7BJY5 137636807 IC50 = 399 nM T68163 CO89DX 137649100 IC50 = 115 nM T68163 CINE03 137652514 IC50 = 1045 nM T68163 C28QUP 137652864 IC50 = 312 nM T68163 CI1D9F 139600335 IC50 = 17 nM T68163 C6VB3O 145925651 IC50 >= 5000 nM T68163 CZ8JC7 145952422 IC50 = 150 nM T68163 CEJ25Z 145955673 IC50 = 9700 nM T68163 C7AIW6 145957749 IC50 = 50 nM T68163 CDA08X 145957845 IC50 = 4200 nM T68163 CF27EG 155511610 IC50 = 2.118 nM T68163 C0AN1O 155512752 IC50 = 644 nM T68163 C2MD1Q 155513187 IC50 > 10000 nM T68163 C3NA2I 155519537 IC50 = 10 nM T68163 CY5MR2 155522337 Ki = 190 nM T68163 C3V4LG 155538413 IC50 = 442 nM T68163 CZQM57 155554194 IC50 = 4297.5 nM T68163 D00ERW 44444843 Ki > 1667 nM T68163 D00HVA 11624601 Ki > 1700 nM T68163 D01IZN 44312289 IC50 > 800000 nM T68163 D02BXJ 46864270 IC50 < 0.15 nM T68163 D02SRA 44312288 IC50 > 800000 nM T68163 D03OKV 9844320 IC50 > 0.5 nM T68163 D04TLI 23657507 IC50 = 1 nM T68163 D05ZUX 44207909 Ki >= 1000 nM T68163 D06HVH 54613583 IC50 > 10000 nM T68163 D06QUQ 5311381 IC50 = 0.4 nM T68163 D06WGX 9549184 IC50 = 1180 nM T68163 D07ERV 44312580 IC50 > 800000 nM T68163 D08RZB 11153014 IC50 = 4 nM T68163 D09DVB 44312287 IC50 > 800000 nM T68163 D0A2LX 44312363 IC50 > 800000 nM T68163 D0B4PI 44312309 IC50 > 800000 nM T68163 D0CE3R 5312137 IC50 = 130 nM T68163 D0H1OK 11562302 Ki = 25.9 nM T68163 D0L4WN 31420 IC50 > 40000 nM T68163 D0OZ2S 11785878 IC50 = 21 nM T68163 D0Q2UZ 44312307 IC50 > 800000 nM T68163 D0Q3NG 11715520 Ki > 1700 nM T68163 D0R2WK 16038120 IC50 = 1308 nM T68163 D0S7IE 11658882 Ki > 1700 nM T68163 D0T2RY 9948320 Ki >= 1000 nM T68163 D0W7LW 44312308 IC50 > 800000 nM T10118 D0K8KX 5280343 IC50 = 100000 nM T10118 D04ZIJ 5478883 IC50 > 100000 nM T10118 D08ZCW 9910174 Ki = 149 nM T10118 D0WY9H 9892148 Ki = 200000 nM T10118 CCFH71 11313 IC50 = 40000 nM T10118 C9Z3SR 17341 IC50 = 25000 nM T10118 C6WXE2 19098 IC50 = 90000 nM T10118 CXEC70 69439 IC50 = 50000 nM T10118 CUJ90R 75195 IC50 = 11000 nM T10118 CEBR78 135053 Ki = 76000 nM T10118 C7RJ0Z 200980 IC50 = 25000 nM T10118 CDB17F 1538822 IC50 = 30000 nM T10118 CNBW97 2250229 IC50 = 27000 nM T10118 C4KO1Z 2799782 IC50 = 2500 nM T10118 C3JU9W 3398697 IC50 = 15000 nM T10118 C57FNV 4422179 IC50 = 80000 nM T10118 CR3NG2 5190983 IC50 = 100000 nM T10118 CJL4X3 5353593 IC50 = 30000 nM T10118 CCT39K 5703472 IC50 = 15000 nM T10118 C1DR3H 6475892 IC50 > 200000 nM T10118 C0MZ5V 6918046 IC50 > 100000 nM T10118 CK64FD 9794516 IC50 > 100000 nM T10118 CKN89B 9822176 Ki > 30000 nM T10118 C7UKF5 9825353 IC50 > 1000 nM T10118 CD5LQ0 9910982 Ki > 15000 nM T10118 CGL12S 9916581 Ki = 458 nM T10118 C0TV8Q 9962561 Ki = 12200 nM T10118 C6ANW0 10004044 Ki = 330000 nM T10118 CHT4F7 10032234 Ki = 34 nM T10118 C8KIA9 10037020 IC50 > 100 nM T10118 C7CW1P 10080504 IC50 = 740 nM T10118 CZH3W7 10094378 Ki = 49000 nM T10118 CD6KX7 10162462 IC50 > 1000 nM T10118 CHVZ36 10251816 IC50 = 950 nM T10118 CKX95D 10257311 Ki = 500 nM T10118 CO3WL8 10347655 Ki = 5800 nM T10118 C9M3VF 10366027 IC50 > 1000 nM T10118 CK2YU1 10369681 Ki = 55 nM T10118 CATB56 10370141 Ki = 720 nM T10118 C2FLG8 10392960 Ki = 9600 nM T10118 CSH83N 10414990 Ki = 6200 nM T10118 CVB41T 10416916 Ki = 364 nM T10118 CWG91R 10472893 Ki > 31000 nM T10118 CKJ46M 10476712 Ki = 2400 nM T10118 C3EN8D 10479280 Ki = 455 nM T10118 C4N9CG 10505462 Ki = 348 nM T10118 C4XU1H 10505893 Ki = 13700 nM T10118 CG1N3Z 10506615 Ki = 1440 nM T10118 C0DV7Q 10528861 Ki = 17900 nM T10118 C5F6RU 10531565 Ki = 1960 nM T10118 CF7A0S 10531953 Ki = 3220 nM T10118 C3UPR0 10554476 Ki = 1830 nM T10118 C8ZXS3 10609754 IC50 > 100 nM T10118 CZ23TH 10627192 Ki = 1630 nM T10118 CH06SV 10627450 Ki = 282 nM T10118 C0TQJ4 10627517 Ki = 3570 nM T10118 CPNI68 10650491 Ki = 177 nM T10118 CBL23T 10674706 Ki = 306 nM T10118 C4FP2G 10674707 Ki = 3280 nM T10118 C2WC3O 10698015 Ki = 1430 nM T10118 C1WV6C 10698103 Ki = 240 nM T10118 C63JIQ 10698344 Ki = 1920 nM T10118 CF1HZ7 10698873 Ki = 780 nM T10118 C04SDQ 10720538 Ki = 27800 nM T10118 CMF61Y 10770047 Ki = 295 nM T10118 CFR3G8 10792830 Ki = 451 nM T10118 CKV52E 10792972 Ki = 171 nM T10118 CUFX71 10793116 Ki = 1400 nM T10118 CEIV70 10793518 Ki = 109 nM T10118 C2D1KY 10820951 IC50 = 37 nM T10118 CSP38Q 11667869 IC50 = 10400 nM T10118 CNK98D 11796320 IC50 = 1000 nM T10118 CKOV89 11799023 Ki = 12.6 nM T10118 C1CQS5 11800896 Ki = 147 nM T10118 CPR4I1 12047383 Ki = 11950 nM T10118 C5U0FJ 12047384 Ki = 384000 nM T10118 C5FU3H 12047385 Ki = 7550 nM T10118 C76QNL 12207594 Ki = 495000 nM T10118 CL54PH 13553439 Ki = 49000 nM T10118 CL1BP2 13615437 Ki = 93000 nM T10118 CUG7D4 13615438 Ki = 112000 nM T10118 COY43I 13615439 Ki = 49000 nM T10118 CAI92R 13615440 Ki = 3900 nM T10118 CW68AF 13615441 Ki = 270 nM T10118 C5L4YZ 13615442 Ki = 1300 nM T10118 CE3IR2 13615444 Ki = 785000 nM T10118 C9J4VU 13615445 Ki = 5600 nM T10118 CZCR18 13615446 Ki = 625000 nM T10118 C8UFN4 13615447 Ki = 63000 nM T10118 CRU13V 13615449 Ki = 1980000 nM T10118 CIA18C 13615450 Ki = 382000 nM T10118 CA7Y2S 13615451 Ki = 267000 nM T10118 C1D5EZ 13615453 Ki = 75000 nM T10118 CV3F2J 13615457 Ki = 927000 nM T10118 C90LWJ 13615458 Ki = 324000 nM T10118 CE0TG3 13660339 Ki = 412000 nM T10118 CU3W9L 13660348 Ki = 470000 nM T10118 CI2Z1C 13660349 Ki = 893000 nM T10118 CB8VK2 13660350 Ki = 1610000 nM T10118 CE0R9C 13660351 Ki = 160000 nM T10118 CF43IW 13660353 Ki = 687000 nM T10118 CK68MB 14542109 Ki > 8000000 nM T10118 CZX4K8 14542110 Ki = 31000 nM T10118 CV1KN9 14799980 IC50 = 200000 nM T10118 CY42MO 15449319 IC50 > 100 nM T10118 CFJB64 15449320 IC50 > 100 nM T10118 C48WFU 15449321 IC50 = 7 nM T10118 CN6M4K 15858923 Ki = 13700 nM T10118 CGHQ54 19697378 IC50 = 10000 nM T10118 C8FB6U 20443937 IC50 = 50000 nM T10118 CDM52L 20443948 IC50 = 15000 nM T10118 C03UHC 20443961 IC50 = 8000 nM T10118 CMR4Z9 20778632 IC50 = 3000 nM T10118 C23OWZ 20778633 IC50 = 13000 nM T10118 CK1C7Q 20778639 IC50 = 700000 nM T10118 CGO1V5 21603623 Ki = 190546.07 nM T10118 C5VSO2 23276168 Ki = 660693.45 nM T10118 CB63KH 23276169 Ki = 501187.23 nM T10118 C7QD8E 23276182 Ki = 707945.78 nM T10118 C0NB6T 44270798 Ki = 295000 nM T10118 C4FY5R 44270803 Ki = 50000 nM T10118 CC9G2D 44286852 Ki = 8400 nM T10118 C0DG5R 44287043 Ki = 4910 nM T10118 C3QD4W 44287797 Ki = 80000 nM T10118 C5W7SA 44287798 Ki = 72000 nM T10118 C02ARM 44287937 Ki > 200000 nM T10118 CP90NM 44288029 Ki = 49000 nM T10118 CRLD46 44292607 IC50 = 9000 nM T10118 CTZR10 44292877 IC50 = 40000 nM T10118 C02ZLR 44292991 IC50 = 15000 nM T10118 CKI80J 44293166 IC50 = 60000 nM T10118 CDUZ42 44293330 IC50 = 2000 nM T10118 CKN8C1 44316486 IC50 = 160 nM T10118 C0YOA6 44331389 IC50 > 100 nM T10118 CGL57V 44331419 IC50 = 70300 nM T10118 C6OPK8 44331423 IC50 > 100000 nM T10118 C5TZL6 44338362 IC50 = 300 nM T10118 C17IOQ 44338363 IC50 = 380 nM T10118 C7UAN4 44338364 IC50 = 420 nM T10118 CWI7N9 44338415 IC50 = 3700 nM T10118 CN05FA 44338434 IC50 = 2100 nM T10118 CXF5Z2 44338508 IC50 = 1900 nM T10118 CBM7L9 44338509 IC50 = 75 nM T10118 CU5H2I 44338658 IC50 > 48000 nM T10118 CC0O3Q 44338659 IC50 > 60000 nM T10118 C09SZK 44338660 IC50 > 60000 nM T10118 CUSP53 44338705 IC50 = 70 nM T10118 C06BSK 44338737 IC50 = 65 nM T10118 CGM1H7 44338738 IC50 = 16000 nM T10118 C4XDT1 44338807 IC50 > 60000 nM T10118 CUFS02 44338809 IC50 = 20000 nM T10118 CZD3L7 44338820 IC50 > 60000 nM T10118 CMK10R 44338821 IC50 > 60000 nM T10118 CP56NM 44338822 IC50 = 280 nM T10118 C6FY8O 44345532 IC50 = 300 nM T10118 C2OH3W 44352031 Ki = 88000 nM T10118 CN5A4R 44381155 Ki = 2900 nM T10118 C6ENF2 44382957 Ki = 92900 nM T10118 CP0YT7 44383405 Ki = 364 nM T10118 CBP42U 44383406 Ki = 1300 nM T10118 C4A5HG 44383407 Ki = 1030 nM T10118 CRGZ24 44383473 Ki = 3950 nM T10118 C03GUY 44383483 Ki > 100000 nM T10118 C9K5XD 44384375 Ki = 1220 nM T10118 CD98YX 44384376 Ki > 100000 nM T10118 CC2LZ6 44384377 Ki = 476 nM T10118 CQ05YV 44384709 IC50 = 38000 nM T10118 CU4O7P 44457950 Ki = 26000 nM T10118 CVI8H9 44459742 Ki = 1090 nM T10118 C0I1KD 53319761 IC50 = 13000 nM T10118 C0WH1K 54675757 Ki = 6309573.44 nM T10118 CL42YZ 54685126 Ki = 223872.11 nM T10118 CJ6BS7 54690337 Ki = 3467368.5 nM T10118 CQ85OF 54694046 Ki = 1819700.86 nM T10118 CV0U6E 54694048 Ki = 549540.87 nM T10118 C95DEC 54694049 Ki = 1348962.88 nM T10118 C9FGL4 54694052 Ki = 691830.97 nM T10118 C01LMD 54694053 Ki = 8128305.16 nM T10118 CL4N6C 54707146 Ki = 79432.82 nM T10118 C28IAV 54732424 Ki = 134896.29 nM T10118 C1T9XJ 54733673 Ki = 512861.38 nM T10118 COA25T 54733674 Ki = 323593.66 nM T10118 CN8Q1F 76333102 IC50 = 40000 nM T10118 CVE7J2 135445689 IC50 = 110000 nM T10118 C5U4IT 135576411 IC50 = 55000 nM T10118 CNL4S3 135843141 IC50 = 220000 nM T10118 D05ICF 3492365 IC50 = 2.4 nM T10118 D07IBU 10696098 IC50 = 70 nM T10118 D0F2YC 10038543 IC50 = 0.69 nM T10118 D0L0QR 443119 Ki = 9.36 nM T10118 D0Q7ST 44338671 IC50 = 50 nM T86161 D02EYG 10096344 IC50 > 100000 nM T86161 D0K8KX 5280343 IC50 = 13000 nM T86161 D0L3DK 6918537 IC50 > 100000 nM T86161 D0NJ5H 11450633 IC50 > 100000 nM T86161 D0R9VR 9651 IC50 > 200000 nM T86161 D0U2JP 4369359 IC50 > 100000 nM T86161 D0W8WB 2353 IC50 = 145000 nM T86161 D07HZG 11516136 IC50 > 30000 nM T86161 D09RJN 9929984 Ki = 1.5 nM T86161 D0FQ2U 6918572 IC50 = 980 nM T86161 D0M3XR 46209133 IC50 > 67000 nM T86161 D05FMP 66561557 IC50 = 4840 nM T86161 D07JHU 71667377 IC50 = 6100 nM T86161 D0C6NX 73356493 IC50 = 1400 nM T86161 D0QX2U 71667229 IC50 = 610 nM T86161 D08PUW 64982 IC50 = 12000 nM T86161 D08RUX 9798234 IC50 = 10 nM T86161 D0A1NU 16049769 Ki > 30000 nM T86161 D0M8AS 195609 IC50 = 3500 nM T86161 C2G5AW 11066 IC50 > 200000 nM T86161 CW8K1N 168928 IC50 = 9750 nM T86161 CF62QN 275182 IC50 > 200000 nM T86161 CHL04T 362574 IC50 = 189000 nM T86161 CKJ1B7 382514 IC50 = 2720 nM T86161 C18OIX 441064 IC50 > 200000 nM T86161 CX08LH 3081017 Ki = 0.97 nM T86161 CIAJ45 3120528 Ki > 30000 nM T86161 CSO4B1 3921011 IC50 = 600 nM T86161 CB7Z3L 6481655 IC50 = 0.5 nM T86161 CNJ0Z3 9800721 Ki > 30000 nM T86161 CM80SI 9801791 IC50 = 2600 nM T86161 CKR9Y5 9823963 IC50 > 100000 nM T86161 CZ1S9O 9942554 IC50 = 61000 nM T86161 C7EV8F 9976844 IC50 = 2.3 nM T86161 C2JDU7 9998765 IC50 = 6.5 nM T86161 C8ECF2 9999371 IC50 = 150 nM T86161 CWU60O 10020162 IC50 = 5.4 nM T86161 CJS28N 10021707 IC50 = 18 nM T86161 C8BYH5 10044551 IC50 = 0.45 nM T86161 CSZ75E 10046311 IC50 > 100000 nM T86161 CZ6QO1 10064965 IC50 = 17 nM T86161 C92BUA 10067693 IC50 = 1.1 nM T86161 C0O1AZ 10088633 IC50 = 91000 nM T86161 CEY8X2 10089498 IC50 = 0.42 nM T86161 CKT8G9 10090257 IC50 = 0.52 nM T86161 CLTR62 10096395 Ki = 0.21 nM T86161 C2H0UF 10149048 IC50 = 1000 nM T86161 CG3O9E 10247989 IC50 = 130 nM T86161 CWU2N1 10339938 IC50 = 0.55 nM T86161 CV5DO6 10340135 IC50 = 0.46 nM T86161 C86BYL 10382642 IC50 = 48 nM T86161 C59GZN 10406121 IC50 = 36 nM T86161 C8D7QV 10406969 IC50 = 1 nM T86161 C5SD4H 10426787 IC50 = 520 nM T86161 CBU0T2 10428014 IC50 = 1.2 nM T86161 C35WMT 10428498 IC50 = 4 nM T86161 CADO92 10428499 IC50 = 38 nM T86161 C4YIR8 10449078 IC50 = 80000 nM T86161 CMI8E7 10449942 IC50 = 94000 nM T86161 C1BJW6 10453899 IC50 = 0.85 nM T86161 CQ4JG2 10545890 IC50 = 11000 nM T86161 CDP3Q0 10570138 IC50 = 2200 nM T86161 CE7I5W 10573308 IC50 = 86 nM T86161 CQ46DO 10614768 IC50 = 30 nM T86161 CWSN46 10622138 IC50 = 1500 nM T86161 C7HZS0 10641689 IC50 > 100000 nM T86161 CL3J9B 10643051 IC50 = 9 nM T86161 C5KPZ9 10662604 IC50 = 23 nM T86161 CLDS86 10671271 IC50 = 5 nM T86161 CHZ87S 10692448 IC50 = 2600 nM T86161 C6D3JS 10736870 IC50 = 50 nM T86161 C05XHR 10737382 IC50 > 100 nM T86161 C1O3RF 10738815 IC50 = 24 nM T86161 CR3MJ8 10781136 IC50 > 100 nM T86161 C2B5NY 10784651 IC50 = 8800 nM T86161 C7Y8SD 10789065 IC50 = 720 nM T86161 C1NW2A 10809317 IC50 = 58 nM T86161 CW4P5M 10810211 IC50 = 40 nM T86161 CV7UJ9 10812075 IC50 = 8000 nM T86161 CO9QM2 11198569 Ki = 0.023 nM T86161 CF1LD8 11199808 Ki = 666 nM T86161 CYL67P 11232890 Ki = 2762 nM T86161 CKL1A8 11268930 Ki = 1741 nM T86161 CM0YI7 11269397 Ki = 925 nM T86161 CEZ27P 11314348 Ki = 40 nM T86161 CW3QZ7 11374531 IC50 > 100000 nM T86161 CL9HN3 11395030 Ki = 245 nM T86161 CTW02K 11406276 Ki = 368 nM T86161 CY15PU 11429829 Ki = 178 nM T86161 CTD0S4 11486251 Ki = 1527 nM T86161 CJV39M 11579395 Ki = 211 nM T86161 C15DLO 11608317 IC50 > 20000 nM T86161 C4KLF3 11740283 IC50 = 24 nM T86161 CM50SP 11742283 IC50 = 1250 nM T86161 C9KI7C 11794456 IC50 = 20 nM T86161 C0P5XM 11794552 IC50 = 17 nM T86161 CE3F9L 11796496 IC50 = 36 nM T86161 CQR35B 11799085 IC50 = 114750 nM T86161 C1BO2L 13889544 IC50 = 14900 nM T86161 CZI1F7 14046925 IC50 = 14000 nM T86161 C7VY1G 14046926 IC50 = 14000 nM T86161 CI3DB4 15951636 IC50 = 1.8 nM T86161 C3SM4T 15951642 IC50 = 10700 nM T86161 C8QRV9 15951839 Ki = 25 nM T86161 CMNT83 15951928 Ki = 191 nM T86161 C13-MAR 16040457 IC50 = 3300 nM T86161 CS7DQ3 16090844 Ki > 30000 nM T86161 C8CVG9 16090856 Ki > 30000 nM T86161 CA1PV5 16216352 IC50 > 20000 nM T86161 C53XZP 16721117 Ki > 30000 nM T86161 CT01PQ 16739331 IC50 > 1000000 nM T86161 CTY8K9 19813462 IC50 = 120 nM T86161 C6ZMS8 21054400 Ki > 30000 nM T86161 C14HFA 21080215 IC50 = 32 nM T86161 CMB0C9 21575462 IC50 = 2866 nM T86161 C0X4SO 22029457 IC50 > 100000 nM T86161 CLK4G6 22029894 IC50 > 100000 nM T86161 C8JSI4 23628284 IC50 > 100000 nM T86161 CU56MV 23643264 IC50 = 15100 nM T86161 C4EG5D 23646512 Ki > 30000 nM T86161 C5GQ7J 23646519 Ki > 30000 nM T86161 CC8JB3 24721570 IC50 = 39740 nM T86161 CSU0B5 25189891 Ki > 30000 nM T86161 CD1UE8 25975470 IC50 = 17 nM T86161 CS40ML 44123747 IC50 > 50000 nM T86161 C5RSX9 44300181 IC50 = 2000 nM T86161 CWLQ89 44305540 IC50 = 3.4 nM T86161 CU2QK6 44305563 IC50 = 8.7 nM T86161 CTR7L6 44305623 IC50 = 60 nM T86161 CVZU70 44305787 IC50 = 510 nM T86161 CZM8K4 44305789 IC50 = 69 nM T86161 C82YKO 44305888 IC50 = 40 nM T86161 CZWI39 44316150 IC50 = 24 nM T86161 CA7N0B 44316393 IC50 = 46 nM T86161 CBMF48 44316461 IC50 = 4.8 nM T86161 CE8L5N 44316588 IC50 = 26 nM T86161 CUW6X5 44316614 IC50 = 50 nM T86161 CIN91J 44316694 IC50 = 5.5 nM T86161 CGJ3D7 44316865 IC50 = 960 nM T86161 CR57NT 44316871 IC50 = 14 nM T86161 C7DA6E 44316872 IC50 = 78 nM T86161 CS76EL 44316886 IC50 = 34 nM T86161 CI92YJ 44316889 IC50 > 100 nM T86161 C2TQ0Z 44316890 IC50 > 100 nM T86161 CPC69K 44316905 IC50 = 27 nM T86161 C8HT0I 44316926 IC50 = 130 nM T86161 CM6QS7 44316928 IC50 = 1400 nM T86161 CSB53A 44316946 IC50 = 150 nM T86161 CD1I0E 44316948 IC50 = 20 nM T86161 C8XE7T 44316949 IC50 > 100 nM T86161 CE7IH5 44329303 Ki = 0.26 nM T86161 C9F5DV 44329392 Ki = 7.5 nM T86161 C2YND3 44329465 Ki = 36 nM T86161 C9GZ6C 44329476 Ki = 0.28 nM T86161 C13DJE 44329488 Ki = 0.34 nM T86161 CW4D7X 44329491 Ki = 0.45 nM T86161 CXN35H 44329692 Ki > 1000 nM T86161 C5BKZ0 44358123 IC50 = 55 nM T86161 CM42ST 44358124 IC50 = 36 nM T86161 C6RM4X 44358125 IC50 = 21 nM T86161 C7E0AK 44358297 IC50 = 14 nM T86161 C7VGO9 44358308 IC50 = 9 nM T86161 CTW19X 44358310 IC50 = 21 nM T86161 CWHZ19 44358311 IC50 = 25 nM T86161 C6JZT1 44358319 IC50 = 54 nM T86161 C2HUO7 44358357 IC50 = 23 nM T86161 C4BMG6 44358443 IC50 = 7 nM T86161 CX8I6C 44381633 IC50 > 100000 nM T86161 CW9F3N 44381634 IC50 > 100000 nM T86161 CI39RJ 44381635 IC50 > 100000 nM T86161 CLK90J 44381645 IC50 > 100000 nM T86161 CT0EO4 44381646 IC50 = 16000 nM T86161 CHX2T7 44381647 IC50 = 27000 nM T86161 C6Y4QW 44381687 IC50 > 100000 nM T86161 CN96MI 44381721 IC50 > 100000 nM T86161 CK4SP1 44381763 IC50 > 100000 nM T86161 CI6RT5 44381811 IC50 > 100000 nM T86161 CG1CD7 44381826 IC50 = 37000 nM T86161 CL51SX 44381845 IC50 = 35000 nM T86161 CXBY42 44381846 IC50 = 59000 nM T86161 C5SV9U 44381847 IC50 = 4200 nM T86161 CRY5K1 44381848 IC50 = 22000 nM T86161 CRE8J7 44381849 IC50 = 19000 nM T86161 CUX2Q9 44381861 IC50 = 77000 nM T86161 C92CKY 44381862 IC50 > 100000 nM T86161 CIX09S 44381884 IC50 > 100000 nM T86161 C3GH0S 44381896 IC50 = 2100 nM T86161 C0FQO1 44381899 IC50 = 1400 nM T86161 CTRX81 44381910 IC50 > 100000 nM T86161 C2XBA5 44381911 IC50 > 100000 nM T86161 CBL60E 44381919 IC50 > 100000 nM T86161 CARK25 44381928 IC50 = 20000 nM T86161 C4LR3K 44381945 IC50 > 100000 nM T86161 CQ4VZ3 44381966 IC50 = 37000 nM T86161 CDCY49 44381967 IC50 > 100000 nM T86161 CT9IN5 44381974 IC50 > 100000 nM T86161 C0FQY4 44381979 IC50 = 29000 nM T86161 CP7XG9 44382005 IC50 > 100000 nM T86161 C6YFP9 44382006 IC50 > 100000 nM T86161 CWJ3V5 44382013 IC50 = 32000 nM T86161 CI8O3F 44382065 IC50 > 100000 nM T86161 CX2JS7 44382077 IC50 = 44000 nM T86161 C38MSH 44382133 IC50 = 40000 nM T86161 C8PD7J 44382134 IC50 = 18000 nM T86161 C89LXF 44382393 IC50 > 100000 nM T86161 CAJ50V 44382443 IC50 > 100000 nM T86161 C8ZP1A 44382444 IC50 = 27000 nM T86161 CKOD04 44382521 IC50 = 76000 nM T86161 CID62U 44418230 Ki = 4.5 nM T86161 CI2H7Q 44418231 Ki = 2.3 nM T86161 CXCV19 44418233 Ki = 2.7 nM T86161 CZW38C 44418239 Ki = 2.2 nM T86161 C7KF0X 44418240 Ki = 53 nM T86161 C8QJ7H 44418242 Ki = 13 nM T86161 C60KPZ 44418243 Ki = 7.4 nM T86161 CMKW39 44418246 Ki = 101 nM T86161 CEBQ24 44418249 Ki = 1359 nM T86161 CVP72G 44418250 IC50 = 130 nM T86161 C59HZQ 44418251 Ki = 2.8 nM T86161 CDX2Q5 44418253 Ki = 1.7 nM T86161 C0RV8O 44418254 Ki = 353 nM T86161 C37KEO 44418255 Ki = 4.4 nM T86161 C08ZST 44440659 Ki > 30000 nM T86161 CR3PM7 44440662 Ki > 30000 nM T86161 CB4Q0H 44440663 Ki > 30000 nM T86161 CCSI57 44440665 Ki > 30000 nM T86161 CF7IS3 44453098 Ki = 6 nM T86161 C3QYD1 44453316 Ki = 16 nM T86161 C32MXK 44458541 IC50 = 700 nM T86161 CZ14DK 44458556 IC50 = 6500 nM T86161 C5VL7T 44458563 IC50 = 420 nM T86161 C8D4WR 44458564 IC50 = 350 nM T86161 CYK8R5 44541222 IC50 = 1400 nM T86161 C6IDA1 44541223 IC50 = 430 nM T86161 C82NWO 44541488 IC50 = 200 nM T86161 C4RS9N 44543393 IC50 = 20 nM T86161 C6F3XA 44543394 IC50 = 3 nM T86161 CRO3D2 44567651 IC50 > 10000 nM T86161 CM95OD 44567652 IC50 > 100000 nM T86161 CX6WL5 44567653 IC50 = 1420 nM T86161 C4MP9D 44567654 IC50 = 9044 nM T86161 CV23FP 44567668 IC50 = 8500 nM T86161 CD4C7Y 44567710 IC50 > 100000 nM T86161 C4CUJ6 44567711 IC50 > 100000 nM T86161 CK1C7W 44567712 IC50 > 10000 nM T86161 CTK1I9 44567713 IC50 = 11790 nM T86161 CM50CU 44567747 IC50 = 14100 nM T86161 CNA0I9 44567918 IC50 = 12300 nM T86161 C6BXT0 44567919 IC50 > 10000 nM T86161 CJ85MG 44567920 IC50 = 9940 nM T86161 CUJD19 44567976 IC50 = 9700 nM T86161 C5YB6E 44567977 IC50 = 392 nM T86161 CNF09E 44567978 IC50 = 26800 nM T86161 C70WEI 44567979 IC50 = 2100 nM T86161 CW7NB6 44568016 IC50 = 492 nM T86161 CY8Z3F 44568017 IC50 = 62200 nM T86161 CRM76D 44568018 IC50 = 18300 nM T86161 CCG83U 44568057 IC50 > 10000 nM T86161 C8XW9A 44568058 IC50 = 417 nM T86161 CMQ7D5 44568097 IC50 > 10000 nM T86161 C1F9OL 44568098 IC50 > 10000 nM T86161 CUYK75 44568099 IC50 > 10000 nM T86161 CZ81XF 44568100 IC50 > 100000 nM T86161 C6GT0A 44568134 IC50 > 10000 nM T86161 C6IW5D 44568135 IC50 = 8700 nM T86161 C3PWD8 44568136 IC50 = 9150 nM T86161 C4NCA7 44568169 IC50 = 46 nM T86161 C8TXH9 44568170 IC50 > 100000 nM T86161 C17PZX 44568171 IC50 > 100000 nM T86161 C7SCJ1 44568172 IC50 > 10000 nM T86161 C60WRN 44575408 IC50 = 57430 nM T86161 CT9W4N 44578393 IC50 = 584 nM T86161 CA57ZD 44578394 IC50 = 53 nM T86161 CTP5L1 44578395 IC50 = 28 nM T86161 CCF86D 44578396 IC50 = 140 nM T86161 CG43QL 44578397 IC50 = 48 nM T86161 CMLW39 44578418 IC50 = 783 nM T86161 CMEL06 44578419 IC50 = 22 nM T86161 CBU72J 44578420 IC50 = 7 nM T86161 C3IUM9 44578421 IC50 = 8 nM T86161 CU8X0T 44578451 IC50 = 28 nM T86161 C6KY5U 44578452 IC50 = 4 nM T86161 CBF82Y 44578453 IC50 = 11 nM T86161 CW0YM2 44578454 IC50 = 270 nM T86161 CMI43H 44578493 IC50 = 343 nM T86161 CQ56RP 44578494 IC50 = 22 nM T86161 CG9PS1 44578495 IC50 = 22 nM T86161 CNDK85 44578496 IC50 = 18 nM T86161 CT8S0X 44578497 IC50 = 64 nM T86161 CGFM25 44578524 IC50 = 34 nM T86161 CTV8N7 44578525 IC50 = 60 nM T86161 CRSD10 44578526 IC50 = 31 nM T86161 CC70DI 44578527 IC50 = 2 nM T86161 CJ0F4L 44578528 IC50 = 3 nM T86161 CR2H9Z 44578556 IC50 = 3100 nM T86161 CDO52N 44578557 IC50 = 1000 nM T86161 CN5VG3 44578558 IC50 = 40 nM T86161 C0YKR1 44578559 IC50 = 34 nM T86161 CE3J7W 44578560 IC50 = 55 nM T86161 CESC37 44578606 IC50 = 43 nM T86161 C5YW7I 44578607 IC50 = 4000 nM T86161 CSEJ25 44578608 IC50 = 2200 nM T86161 CBFY24 44578609 IC50 = 800 nM T86161 CAV68C 44578610 IC50 = 900 nM T86161 C6DH7S 44578642 IC50 = 70 nM T86161 C84UYL 44578643 IC50 = 250 nM T86161 C9AD1Z 44578644 IC50 = 40 nM T86161 CG26FT 44578645 IC50 = 30 nM T86161 C4UFW2 44578646 IC50 = 80 nM T86161 CZ8W0G 44578681 IC50 = 12 nM T86161 CM50QV 44578682 IC50 = 17 nM T86161 CN38WL 44578683 IC50 = 15 nM T86161 CB6GM1 44584127 IC50 = 1400 nM T86161 CXYT36 45101723 IC50 > 100000 nM T86161 C2RNP7 45102670 IC50 > 100000 nM T86161 C28ZXW 45487888 IC50 = 39000 nM T86161 C2N3IZ 45487894 IC50 > 100000 nM T86161 CP62TC 45487898 IC50 = 48000 nM T86161 CWQ1R9 45487903 IC50 = 61000 nM T86161 C8H1KY 45487904 IC50 > 100000 nM T86161 C6X7WJ 45487908 IC50 > 100000 nM T86161 C5OXM9 45487915 IC50 > 100000 nM T86161 CPJ19X 45487917 IC50 > 100000 nM T86161 CV2R7M 45487920 IC50 = 43000 nM T86161 C57JRG 45487921 IC50 = 33000 nM T86161 C4JD1P 45487922 IC50 > 100000 nM T86161 CPB85R 45487926 IC50 = 45000 nM T86161 CTY16E 45487930 IC50 = 57000 nM T86161 C4QTL9 45487931 IC50 = 65000 nM T86161 CG9V0L 45487940 IC50 = 72000 nM T86161 C5XTV1 45487945 IC50 = 15000 nM T86161 C3VK4G 45487946 IC50 > 100000 nM T86161 COBY30 46231131 IC50 = 5.6 ug.mL-1 T86161 CLE0Y4 46889276 IC50 = 65000 nM T86161 CBE93O 46889313 Ki = 5540 nM T86161 CHT91Q 46898083 IC50 = 26 nM T86161 CS5X9L 46917048 IC50 > 100000 nM T86161 C80RAT 47370344 IC50 > 100000 nM T86161 CI6QC3 49795929 IC50 = 89000 nM T86161 CZ7A9E 49796933 IC50 = 100000 nM T86161 C5RF0Y 49796938 IC50 > 100000 nM T86161 C8WYA5 49796953 IC50 = 39000 nM T86161 CQH86V 49796955 IC50 > 100000 nM T86161 CN12AO 53353383 IC50 = 31600 nM T86161 C51GUC 53354365 IC50 > 100000 nM T86161 CRJ5P9 53354369 IC50 > 100000 nM T86161 C4G2HT 53354470 IC50 > 100000 nM T86161 C8GPO1 56665883 IC50 = 6000 nM T86161 C4AY5G 60195086 IC50 < 50 nM T86161 CIY07P 60195087 Ki = 23 nM T86161 CB9E2P 60195088 Ki = 160 nM T86161 CW64RD 66561555 IC50 = 1100 nM T86161 C9GTI7 66561556 IC50 > 10000 nM T86161 CLO96S 70681357 IC50 = 5800 nM T86161 CWP41T 70681469 IC50 = 15900 nM T86161 C7Z2KY 70681470 IC50 = 9400 nM T86161 C19XIQ 70683454 IC50 = 1600 nM T86161 C07ADL 70683455 IC50 > 100000 nM T86161 CO2NK6 70685557 IC50 = 2600 nM T86161 CK0WX8 70685558 IC50 = 600 nM T86161 CLF84U 70685559 IC50 > 50000 nM T86161 C0K7PS 70685560 IC50 > 100000 nM T86161 C2T0NS 70685696 IC50 = 6 nM T86161 CVD76F 70687705 IC50 > 100000 nM T86161 C28GVW 70687706 IC50 > 50000 nM T86161 CUY81P 70689750 IC50 > 10000 nM T86161 CX2O0Z 70689751 IC50 > 100000 nM T86161 C17YKW 70689752 IC50 > 100000 nM T86161 C87LMG 70691901 IC50 = 5400 nM T86161 CL5EG7 70691902 IC50 > 50000 nM T86161 CGND49 70691903 IC50 > 100000 nM T86161 CGT57B 70691904 IC50 > 100000 nM T86161 CT89CW 70691905 IC50 > 100000 nM T86161 C5WI6V 70691906 IC50 > 100000 nM T86161 CQMV53 70693949 IC50 = 2900 nM T86161 CBP8U7 70693950 IC50 > 10000 nM T86161 C0I2CV 70693951 IC50 > 10000 nM T86161 CCB64G 70693952 IC50 > 50000 nM T86161 C3ZUK2 70693953 IC50 > 50000 nM T86161 CS76EN 70693954 IC50 > 100000 nM T86161 C27PFC 70693955 IC50 > 100000 nM T86161 CVY48R 70693956 IC50 > 100000 nM T86161 CA01KO 70696068 IC50 = 5000 nM T86161 CSW43K 70696069 IC50 = 1700 nM T86161 C7B8AO 71621488 IC50 > 1800 nM T86161 C8T2PW 71655265 IC50 = 5 nM T86161 C1HGS0 71655267 IC50 = 1800 nM T86161 C9XJ6S 71655268 IC50 = 91000 nM T86161 CX6AI5 71655326 IC50 = 640 nM T86161 C9H0QK 71655327 IC50 = 2100 nM T86161 CLM0G6 71655328 IC50 = 1300 nM T86161 CFS59P 71655329 IC50 = 1000 nM T86161 CZL7N9 71655330 IC50 = 440 nM T86161 CR7I0Y 71655331 IC50 = 26 nM T86161 CLCH69 71655332 IC50 = 96 nM T86161 CL0ZS6 71655390 IC50 = 1600 nM T86161 C6Y9LQ 71655391 IC50 = 320 nM T86161 C93CXQ 71655392 IC50 = 110 nM T86161 C8P1GB 71655393 IC50 = 57 nM T86161 CVB75Q 71655394 IC50 = 1.8 nM T86161 CH4ZS0 71655395 Ki = 0.73 nM T86161 CC93KJ 71655554 IC50 = 860 nM T86161 CN90KH 71655555 IC50 = 13200 nM T86161 CUT37D 71655556 IC50 = 53600 nM T86161 C71OFQ 71655557 IC50 = 1000 nM T86161 C7R6HU 71655622 IC50 = 16800 nM T86161 C2NA1M 71655623 IC50 > 50000 nM T86161 CDF08H 71655624 IC50 = 610 nM T86161 CBEX27 71655625 IC50 = 3400 nM T86161 CT6XB5 71655626 IC50 = 2400 nM T86161 C1ND2P 71655627 IC50 = 11700 nM T86161 CXZ8N4 71667081 IC50 = 640 nM T86161 CJ9QU7 71667226 IC50 = 11300 nM T86161 CE0Z8G 71667227 IC50 = 8200 nM T86161 CL7CS3 71667230 IC50 = 840 nM T86161 CB6SI5 71667231 IC50 = 710 nM T86161 C75UWV 71667375 IC50 = 350 nM T86161 C19CTI 71667376 IC50 = 360 nM T86161 C69CJB 71667378 IC50 = 1200 nM T86161 C07HNK 71667379 IC50 = 11800 nM T86161 CK74SP 71667380 IC50 = 29100 nM T86161 CMYZ68 71667381 IC50 = 7200 nM T86161 CDI39U 71667510 IC50 = 13700 nM T86161 CC10AZ 73345857 IC50 > 50000 nM T86161 CX4F0Y 73347359 IC50 = 18500 nM T86161 C3XFM5 73347360 IC50 = 38000 nM T86161 CR09PJ 73348871 IC50 = 2400 nM T86161 C06WRM 73350448 IC50 > 100000 nM T86161 C1T7LK 73350449 IC50 = 7700 nM T86161 CCIZ12 73350450 IC50 = 5600 nM T86161 CFV5U3 73353424 IC50 = 33000 nM T86161 CRS4O0 73353425 IC50 = 8300 nM T86161 CLYP23 73354936 IC50 = 350 nM T86161 CMC5A1 73356072 IC50 = 5.5 nM T86161 CH9W2R 73356494 IC50 = 600 nM T86161 CKD46T 73356495 IC50 > 100000 nM T86161 CI0N6E 73356496 IC50 = 39000 nM T86161 CL43XA 86302389 IC50 = 15200 nM T86161 CIV7Y8 89668929 IC50 > 100000 nM T86161 C87GJT 89704940 IC50 > 100000 nM T86161 CHI7U9 89704942 IC50 = 5900 nM T86161 CSLI09 89704955 IC50 > 100000 nM T86161 CA3K7R 89704970 IC50 = 8700 nM T86161 CF89OD 89705045 IC50 = 2000 nM T86161 CK3Z8J 89705076 IC50 > 100000 nM T86161 CH6P0S 89705081 IC50 = 500 nM T86161 C63DGS 89705096 IC50 = 9100 nM T86161 CND56S 89705098 IC50 = 24000 nM T86161 C0CKQ7 89705100 IC50 = 2030 nM T86161 C0CPD1 89705103 IC50 = 3400 nM T86161 C1IL7N 89705109 IC50 = 11.2 nM T86161 CA48MR 89705136 IC50 = 2700 nM T86161 C5F9OA 89705152 IC50 = 9300 nM T86161 C1VSG5 89705179 IC50 = 22000 nM T86161 CHAS49 89705195 IC50 = 14200 nM T86161 C0RP1J 89705223 IC50 = 6600 nM T86161 CQO0I6 89705242 IC50 = 5800 nM T86161 C7DF1P 89705244 IC50 = 1280 nM T86161 C03OGJ 89705273 IC50 = 19400 nM T86161 CGX4I7 89705275 IC50 = 8300 nM T86161 CX9BC3 89712515 IC50 > 100000 nM T86161 C6TGZ5 90655538 IC50 = 44 nM T86161 C9P3HJ 90655539 IC50 = 46000 nM T86161 CT98OM 90655540 IC50 = 25000 nM T86161 CVQ8M4 90655541 IC50 = 2600 nM T86161 CT6Q2L 90655542 IC50 = 9000 nM T86161 C7Z4GV 90655543 IC50 = 6300 nM T86161 CE3HC2 90655544 IC50 = 2000 nM T86161 CU2I3V 90655545 IC50 > 50000 nM T86161 C2NZ7X 90655546 IC50 > 25000 nM T86161 C0E5UP 90655547 IC50 = 67000 nM T86161 CF23RI 90655548 IC50 > 100000 nM T86161 CW3QG7 90655549 IC50 > 100000 nM T86161 CHG4E2 90655550 IC50 > 100000 nM T86161 CTA78W 90655551 IC50 = 9000 nM T86161 CA6S4W 90655552 IC50 = 6800 nM T86161 C3LT0S 90655553 IC50 = 7300 nM T86161 CEW45X 90655554 IC50 = 33700 nM T86161 CRX52D 90655555 IC50 = 39000 nM T86161 C9KG1U 90655556 IC50 = 48000 nM T86161 CXYE76 90655557 IC50 = 5600 nM T86161 CES85Q 90655558 IC50 > 100000 nM T86161 CK7IB9 90655559 IC50 = 290 nM T86161 CAG5X4 90655560 IC50 > 100000 nM T86161 C3IJA0 90655561 IC50 > 50000 nM T86161 C4V0ZY 90655562 IC50 = 780 nM T86161 CY9G8Q 90655563 IC50 = 16800 nM T86161 CV0SF5 90664925 IC50 > 10000 nM T86161 C37EPA 90666507 IC50 = 75000 nM T86161 CM7E4V 101887269 IC50 > 100000 nM T86161 C8EH0J 101887270 IC50 > 100000 nM T86161 CDT67J 101887271 IC50 > 100000 nM T86161 C4F2CS 101887272 IC50 > 100000 nM T86161 C58XWA 101887273 IC50 > 100000 nM T86161 C3Y9ET 101887274 IC50 > 100000 nM T86161 C1AF8C 101887275 IC50 > 100000 nM T86161 CH7QC5 101887276 IC50 > 100000 nM T86161 CO4FR2 101887277 IC50 > 100000 nM T86161 C9JEH0 101887278 IC50 > 100000 nM T86161 C52GIO 101887279 IC50 > 100000 nM T86161 CGT0U7 118707566 IC50 > 50000 nM T86161 CI38CB 118707567 IC50 > 50000 nM T86161 CR24BC 118707568 IC50 = 11500 nM T86161 CWF49N 118707569 IC50 > 50000 nM T86161 C8PQ7A 118707570 IC50 = 17700 nM T86161 CJ62AB 118707571 IC50 = 3500 nM T86161 C0ZP2V 122179016 IC50 = 27.8 ug.mL-1 T86161 CN78TQ 122189864 IC50 > 100000 nM T86161 CNM82F 122189865 IC50 > 100000 nM T86161 C19GHJ 122189866 IC50 > 100000 nM T86161 C3U9KC 122189867 IC50 > 100000 nM T86161 CW5V3U 122189868 IC50 > 100000 nM T86161 CCG05R 122189869 IC50 > 100000 nM T86161 CI01PT 122189870 IC50 > 100000 nM T86161 C80EWF 122189871 IC50 > 100000 nM T86161 C3N7JC 122189872 IC50 > 100000 nM T86161 CG8O1J 122189873 IC50 > 100000 nM T86161 CK0US2 122189874 IC50 > 100000 nM T86161 C5V6NI 122189875 IC50 > 100000 nM T86161 CV7A9Y 122189876 IC50 > 100000 nM T86161 CH97SN 122189877 IC50 > 100000 nM T86161 CN86VR 122189878 IC50 > 100000 nM T86161 CZB49I 122189879 IC50 > 100000 nM T86161 CUTO40 127050021 Ki = 10 nM T86161 C8FOA6 127050022 Ki = 0.75 nM T86161 C2FA9N 127050023 Ki = 46 nM T86161 CV2F8G 127050024 Ki = 80000 nM T86161 CZE76Y 127050075 Ki > 150000 nM T86161 C5SE9N 127050076 Ki = 12000 nM T86161 CND8J7 127050077 Ki = 67000 nM T86161 CO2P4U 127050078 Ki = 65000 nM T86161 C80DBR 127050315 Ki > 150000 nM T86161 CE96SX 127050612 Ki = 7500 nM T86161 CS97OM 127050628 Ki = 32.5 nM T86161 CPA24W 127050629 Ki = 1000 nM T86161 CYA42B 127050630 Ki = 1500 nM T86161 CTB76I 127050631 Ki = 62500 nM T86161 CDC0R1 127050945 Ki > 150000 nM T86161 CN2O4A 127050949 Ki = 4000 nM T86161 C9O7PK 127051276 Ki > 150000 nM T86161 C4AKL1 127051277 Ki = 2100 nM T86161 C4CWL6 127051278 Ki = 62000 nM T86161 CY1O5Q 145967090 IC50 = 950 nM T86161 C9IK2U 155510659 Ki = 210 nM T86161 C5LP2Z 155512771 Ki = 290 nM T86161 CJ7NB0 155512973 Ki = 355 nM T86161 C1J9YK 155514168 Ki = 11400 nM T86161 CHK67A 155515001 Ki = 6300 nM T86161 CCX7H6 155521556 Ki = 270 nM T86161 CK5YZ8 155521752 Ki = 3.5 nM T86161 CZ23TD 155522229 Ki = 1100 nM T86161 CE58QC 155522835 Ki = 1000 nM T86161 CE8S1P 155523369 Ki > 100000 nM T86161 CC0JR7 155523397 Ki = 767 nM T86161 CHFS52 155524138 Ki > 15000 nM T86161 CAYB79 155525876 Ki > 15000 nM T86161 CVEX75 155528980 Ki = 170 nM T86161 C8EQ4C 155530631 IC50 = 1.3 nM T86161 C8JC7P 155533583 Ki > 30000 nM T86161 CPB6J5 155536851 Ki = 49 nM T86161 CV4Y6F 155537130 Ki = 3300 nM T86161 CC6Y5D 155545709 Ki = 80 nM T86161 CR0NB1 155545817 Ki = 3000 nM T86161 CN1H6W 155545965 Ki = 950 nM T86161 CVT78K 155553875 Ki = 9 nM T86161 C3OVS2 155557727 Ki = 22 nM T86161 CH5E6R 155557938 Ki = 6 nM T86161 C5BXI4 155565399 Ki = 44 nM T86161 CAZ87J 155565932 Ki = 620 nM T86161 CWPL14 155566983 IC50 > 200000 nM T86161 CU6TM7 155567204 Ki = 2200 nM T86161 CG3BR0 155567943 IC50 = 67000 nM T86161 D00YEV 5281605 IC50 = 36000 nM T86161 D02SGJ 19009 IC50 > 200000 nM T86161 D02XEX 11168203 IC50 = 7890 nM T86161 D03DNV 71655266 IC50 = 990 nM T86161 D04CAR 10607286 IC50 = 47000 nM T86161 D06FNK 122623 Ki = 0.4 nM T86161 D09ALJ 5280805 IC50 > 200000 nM T86161 D09VYW 9847548 IC50 = 36320 nM T86161 D0G3TK 5280863 IC50 > 200000 nM T86161 D0JL2T 5393152 IC50 > 200000 nM T31204 D00JVR 2267 Ki = 19.95 nM T31204 D00XWD 135409453 Ki < 1.995 nM T31204 D01AZG 5073 Ki = 19.95 nM T31204 D01JMC 11658860 Ki = 1.3 nM T31204 D01XBA 5035 Ki = 69 nM T31204 D01ZII 2726 Ki = 39.81 nM T31204 D03ELL 2159 Ki = 316.23 nM T31204 D04EGX 54746 Ki = 1.4 nM T31204 D04JEE 4946 EC50 > 5011.87 nM T31204 D05AHE 8226 Ki = 0.8 nM T31204 D06FES 667477 Ki = 25.3 nM T31204 D06XZR 27400 Ki = 2 nM T31204 D08VRO 3822 Ki = 180 nM T31204 D0CQ0Z 33630 Ki = 184 nM T31204 D0H3HM 60795 Ki = 0.36 nM T31204 D0H7KF 5002 Ki = 251.19 nM T31204 D0O6GC 9681 Ki = 7.586 nM T31204 D0P0OU 11978813 Ki = 0.3981 nM T31204 D0R1JV 60854 Ki = 1.585 nM T31204 D0U5FS 3396 Ki = 151.4 nM T31204 D0V4QS 135398745 Ki = 6.31 nM T31204 D0W5HK 216239 Ki = 56 nM T31204 D0YG7M 3827 Ki = 31.62 nM T31204 D0Z1RV 135398737 Ki = 3.162 nM T31204 D01HLO 58438464 IC50 = 3700 nM T31204 D04GMY 11842633 Ki < 1.995 nM T31204 D0HZ2E 5311271 Ki = 1258.93 nM T31204 D0LI1C 44469321 IC50 > 10000 nM T31204 D0R9KG 11604525 Ki > 10000 nM T31204 D0U0KR 3035850 Ki = 2770 nM T31204 D0W4XY 11502243 Ki = 3.4 nM T31204 D0Y6ZK 123683 Ki = 1080 nM T31204 D0I5VA 11248240 IC50 = 3260 nM T31204 D02FEA 3336 Ki = 3217 nM T31204 D02JMI 9888211 Ki = 1.585 nM T31204 D03YPJ 5163 Ki = 4.3 nM T31204 D03ZZH 9887537 Ki = 12.59 nM T31204 D04DGE 9888804 Ki = 31.62 nM T31204 D06ZVC 10150497 Ki = 458 nM T31204 D08AWI 11430856 Ki > 5000 nM T31204 D08NLQ 114709 Ki > 10000 nM T31204 D0B4BN 3045227 EC50 = 1.585 nM T31204 D0B7SP 11292933 Ki = 501.19 nM T31204 D0EE6L 3038495 Ki = 33.1 nM T31204 D0M7LV 5761 Ki = 30 nM T31204 D0Q2JS 10436045 Ki = 25.12 nM T31204 D0QF4Z 196968 IC50 = 0.7 nM T31204 D0S5FQ 7153 EC50 = 93 nM T31204 D0U7VZ 11225102 Ki < 1.995 nM T31204 D0YP7L 6604889 Ki = 5 nM T31204 C7B8VJ 44405080 Ki = 12 nM T31204 CZUI83 2769 Ki = 39.81 nM T31204 C5H9CN 9287 EC50 = 75.8 nM T31204 C6KIN7 10624 EC50 = 74 nM T31204 CFGH18 27620 Ki = 614 nM T31204 CR69PX 29101 Ki = 5500 nM T31204 C4RF5C 30241 Ki = 8.3 nM T31204 CF3R1X 38240 Ki = 555.1 nM T31204 CN9GK1 104911 Ki = 24 nM T31204 CD6Y4C 126769 Ki = 21 nM T31204 CLK7P3 169713 IC50 = 54 nM T31204 C2V5FA 398712 Ki = 53 nM T31204 CA7NP1 732268 Ki = 151.3 nM T31204 C2VLP8 752521 Ki = 20.5 nM T31204 C7I9SV 752565 IC50 = 1056 nM T31204 CDK19P 879244 Ki = 19.8 nM T31204 CQ8TV4 895660 IC50 = 280 nM T31204 C9JN8C 1082900 IC50 > 6500 nM T31204 CYE02G 1400243 EC50 < 10000 nM T31204 C2VK3F 1430062 IC50 > 13000 nM T31204 CC1M8I 1452981 IC50 > 10000 nM T31204 CS7KJ5 2267399 IC50 = 485.9 nM T31204 CPI2C5 2775690 Ki = 407 nM T31204 CF7E4X 2884131 Ki = 53.3 nM T31204 CJ6D8N 3342390 Ki < 1000 nM T31204 C7W1FS 3391669 IC50 = 542 nM T31204 CGLB95 3400827 IC50 = 791 nM T31204 CV1WY3 3410378 IC50 = 5000 nM T31204 CEO5I1 3442850 IC50 = 92 nM T31204 CHI1W6 3465057 IC50 > 10000 nM T31204 CN9AF5 3473601 IC50 = 753 nM T31204 C2I3OU 3499360 IC50 = 856 nM T31204 C3HJK8 3525815 IC50 = 1600 nM T31204 CS8KE2 3649661 Ki = 7.2 nM T31204 CEHA49 3716424 IC50 = 175 nM T31204 CK9T8C 3723094 IC50 = 30 nM T31204 CZ9U1L 3735585 IC50 < 10 nM T31204 C1VCM9 3736302 IC50 = 188 nM T31204 CL6UY1 3743171 IC50 = 100 nM T31204 C5YQ9W 3751272 IC50 = 350 nM T31204 C2FU3V 3757038 IC50 = 5000 nM T31204 CLVJ27 3765560 IC50 = 426 nM T31204 C3T5RZ 3773677 IC50 = 5000 nM T31204 C0KEL4 3777203 IC50 < 10 nM T31204 CH36OS 3781561 IC50 = 1281 nM T31204 CW3VP0 3802375 IC50 = 5000 nM T31204 CBI1D7 3826158 IC50 = 179 nM T31204 CX87FY 3830738 IC50 = 133 nM T31204 CYPH98 3845148 Ki = 310 nM T31204 CQ8IV6 3898525 IC50 = 15 nM T31204 CWYC34 4148445 IC50 = 531 nM T31204 CI67XC 4203621 IC50 = 1470 nM T31204 C1SQ5X 4297073 IC50 = 42 nM T31204 C3D2GH 4322819 IC50 = 46 nM T31204 CF1DO7 4366334 IC50 = 1.8 nM T31204 CQ03WP 4518239 IC50 = 427 nM T31204 CMTG46 4601219 IC50 > 10000 nM T31204 CYT32E 4657811 IC50 = 5000 nM T31204 CF7DH2 4679720 IC50 = 5000 nM T31204 C4X9MT 4895014 IC50 = 95 nM T31204 CW2C1I 5009938 Ki = 497 nM T31204 CT3F1S 5093797 IC50 = 280 nM T31204 CA68EI 5113614 IC50 = 29 nM T31204 C4OD9L 5128094 IC50 = 50 nM T31204 CHF83G 5165122 IC50 = 5000 nM T31204 CS10EQ 5167627 IC50 = 500 nM T31204 CY67TC 5281073 Ki = 1.9 nM T31204 CAO47E 6452095 Ki = 87 nM T31204 C0QCK1 6918455 Ki < 3981.07 nM T31204 C1WXY3 6918603 Ki < 5011.87 nM T31204 CD0Z4I 6918648 Ki = 1000 nM T31204 CB5A6I 9799300 Ki < 1584.89 nM T31204 CE0DI5 9804612 Ki < 7943.28 nM T31204 CNX4F0 9805456 Ki < 6309.57 nM T31204 C0H6DZ 9837204 Ki = 221 nM T31204 C28HIY 9839057 Ki = 0.19 nM T31204 C7H8CZ 9839920 Ki = 2.512 nM T31204 CDOC72 9844378 Ki > 10000 nM T31204 CM13ZV 9856041 Ki = 13 nM T31204 CKQ5O7 9856509 Ki = 25 nM T31204 C9B2QD 9859144 Ki = 53 nM T31204 C0ZR3E 9861687 IC50 = 9.772 nM T31204 C0W3JF 9866423 Ki = 501.19 nM T31204 C19KGY 9869628 Ki = 125.89 nM T31204 C7AB8O 9870053 Ki < 3981.07 nM T31204 C2ELZ9 9881053 IC50 = 200 nM T31204 CKS8Z9 9881119 EC50 = 36 nM T31204 CE46QD 9881885 EC50 = 100 nM T31204 CJW1P5 9888494 Ki = 1000 nM T31204 C6N8UE 9889681 Ki < 7943.28 nM T31204 CM52WU 9890119 Ki < 5011.87 nM T31204 CEG1K5 9891002 Ki = 1258.93 nM T31204 C7QMK5 9891617 Ki < 7943.28 nM T31204 CEL29O 9891618 Ki < 10000 nM T31204 C3J8GU 9892409 Ki = 1995.26 nM T31204 C2P3GS 9899500 Ki = 19 nM T31204 CYWQ50 9906447 Ki = 3152 nM T31204 CYZ5N4 9909089 Ki = 316.23 nM T31204 CO7BK6 9909648 Ki = 69.6 nM T31204 C78MDV 9913554 Ki = 1258.93 nM T31204 C6BTZ9 9920815 Ki = 13 nM T31204 CR9KM0 9921064 Ki = 245 nM T31204 CO6MD4 9931534 Ki = 7.943 nM T31204 C4L1GA 9934033 IC50 = 9.66 nM T31204 CYVZ47 9934284 Ki = 1000 nM T31204 CWO45F 9935387 Ki = 1258.93 nM T31204 CYH3R7 9947817 Ki > 10000 nM T31204 CK8NR2 9954121 Ki < 5011.87 nM T31204 CFR41N 9957068 Ki < 1000 nM T31204 CFN50J 9978683 Ki = 601 nM T31204 C76JBU 9981505 Ki < 398.11 nM T31204 C2USG0 9983031 Ki < 1000 nM T31204 CL9UJ7 9990808 EC50 = 316.23 nM T31204 C9FBE5 9991444 EC50 = 50.12 nM T31204 C7P2BT 9994008 EC50 = 40 nM T31204 CYG36Z 10003368 Ki < 1584.89 nM T31204 CT2CS3 10003477 Ki < 1584.89 nM T31204 C3C0YF 10008294 Ki = 1258.93 nM T31204 CLE61D 10015414 EC50 = 130 nM T31204 C45HCE 10017554 Ki = 1.15 nM T31204 CEY30Z 10017556 EC50 = 230 nM T31204 CK18LT 10020895 Ki > 10000 nM T31204 C12LON 10036629 EC50 = 63.1 nM T31204 C2ZO8M 10037962 Ki > 5000 nM T31204 C25WVJ 10047566 IC50 > 1000 nM T31204 C6M1TH 10050022 Ki = 398.11 nM T31204 CDSQ03 10058473 Ki = 483 nM T31204 C5PG9D 10064386 EC50 = 64 nM T31204 CD2RM6 10085260 Ki = 255 nM T31204 CC5IZ2 10103618 Ki = 58.5 nM T31204 C8F9SD 10105208 EC50 = 380 nM T31204 CJ1K5Y 10127939 Ki = 79.43 nM T31204 CZ2S7U 10127968 Ki = 125.89 nM T31204 C8ZJ9G 10131066 Ki = 11 nM T31204 CJF76C 10150393 Ki = 1584.89 nM T31204 CI2X3Y 10151289 Ki = 158.49 nM T31204 CN78BA 10176869 Ki = 140 nM T31204 CUJ06B 10194524 Ki = 794.33 nM T31204 C02TKP 10216639 Ki > 7943.28 nM T31204 CRNG42 10217207 Ki = 316.23 nM T31204 C96ARE 10217208 Ki = 1258.93 nM T31204 CRJ01O 10237852 Ki = 1995.26 nM T31204 C21CDB 10244831 Ki = 31.62 nM T31204 C4Q2SH 10249573 Ki = 1995.26 nM T31204 CKT7U9 10254433 Ki < 501.19 nM T31204 CD27VE 10255548 Ki = 39.81 nM T31204 CMRA02 10257042 Ki = 501.19 nM T31204 COAP98 10287912 Ki = 63 nM T31204 CAT4H3 10288601 Ki = 316.23 nM T31204 CPW71K 10309622 Ki = 1258.93 nM T31204 CFWC08 10321945 Ki < 630.96 nM T31204 CRT0J7 10329912 EC50 > 10000 nM T31204 CE07JM 10330266 Ki = 214 nM T31204 CT4L5Z 10331841 EC50 = 1500 nM T31204 C9IAV3 10346043 Ki > 3162.28 nM T31204 C86INY 10346749 Ki = 199.53 nM T31204 CS24DU 10353268 Ki = 14 nM T31204 CBQ57F 10368126 Ki = 794.33 nM T31204 CC1GT2 10368204 Ki = 251.19 nM T31204 C23KXL 10371119 Ki = 1258.93 nM T31204 CV2G9H 10379910 EC50 = 1000 nM T31204 CMZA83 10383646 Ki = 978 nM T31204 C36BOF 10389430 IC50 = 442 nM T31204 C1R5GY 10390089 Ki = 199.53 nM T31204 CA3NO7 10401602 EC50 = 180 nM T31204 C0ON1Z 10408409 Ki = 158.49 nM T31204 CYA49X 10409431 Ki < 794.33 nM T31204 C5PCO9 10410103 Ki < 10000 nM T31204 CK6G0O 10413268 Ki = 158.49 nM T31204 C4TPN1 10413595 Ki = 630.96 nM T31204 C2B0IU 10421236 Ki = 150 nM T31204 CR4LS0 10430623 Ki = 236 nM T31204 CD7U5I 10433930 Ki = 1995.26 nM T31204 CNJ4Z9 10435572 Ki = 31.62 nM T31204 C8TSH1 10454231 Ki = 501.19 nM T31204 CA43RM 10457586 Ki < 10000 nM T31204 CSV35T 10458193 Ki = 63.1 nM T31204 C2QO7W 10458785 Ki = 199.53 nM T31204 CTED07 10465263 EC50 = 1000 nM T31204 COV85C 10472143 Ki = 27 nM T31204 CRG9T1 10472780 EC50 > 10000 nM T31204 CS01JP 10476876 Ki = 630.96 nM T31204 CX13YD 10477339 Ki < 1995.26 nM T31204 C12RUZ 10479309 Ki = 1584.89 nM T31204 CH64LD 10479409 Ki = 125.89 nM T31204 CQA0U8 10503674 Ki = 100 nM T31204 CRK20I 10526616 Ki = 19.95 nM T31204 CNU6K9 10527432 Ki = 5.012 nM T31204 C4EN0P 10528314 Ki = 39.81 nM T31204 CKG7E2 10541003 Ki = 11200 nM T31204 CMGY61 10549658 Ki = 12.59 nM T31204 CBU41F 10550405 Ki = 5.012 nM T31204 C0PV1R 10550406 Ki = 15.85 nM T31204 C2A6FZ 10568771 Ki = 1.15 nM T31204 C9NQK8 10573762 Ki = 10 nM T31204 CHE80N 10573876 Ki < 1584.89 nM T31204 C4WGZ3 10574607 Ki = 25.12 nM T31204 CO23YX 10597140 Ki = 3981.07 nM T31204 C2O3BC 10599545 Ki = 25.12 nM T31204 CAG6B7 10609802 Ki = 205 nM T31204 CVKA91 10622480 Ki = 7.943 nM T31204 CW8YO5 10623020 Ki = 3.981 nM T31204 CYT8G2 10623205 Ki = 7.943 nM T31204 C38YWE 10670191 Ki = 6.31 nM T31204 CJC59K 10670813 Ki = 10 nM T31204 C7BJO5 10690185 Ki = 3.981 nM T31204 C7QZO5 10693974 Ki = 63.1 nM T31204 CY3MJ1 10714852 Ki = 15.85 nM T31204 CJR6Y5 10718089 Ki = 15.85 nM T31204 CQ95BN 10740494 Ki = 10 nM T31204 CE5U6G 10740495 Ki = 10 nM T31204 C49CTY 10741816 Ki = 12.59 nM T31204 C7H8VX 10751567 Ki = 311 nM T31204 CBUA63 10764263 Ki = 10 nM T31204 C26JIN 10767350 Ki = 15.85 nM T31204 CF2R3P 10791286 Ki = 19.95 nM T31204 CG5B6Z 10808965 Ki = 10 nM T31204 CT65RQ 10811153 Ki = 31.62 nM T31204 CUD58N 10812577 Ki = 1995.26 nM T31204 CKU7G0 10813396 Ki = 501.19 nM T31204 CPXC32 10830245 Ki = 158.49 nM T31204 C8MHZ9 10835110 Ki < 1000 nM T31204 C5AI2P 10835537 Ki = 25.12 nM T31204 CFE3J6 10835585 Ki = 398.11 nM T31204 CGX81B 10837002 Ki = 50.12 nM T31204 CL3XI5 10837468 Ki = 7.943 nM T31204 CCJ9Y2 10898996 EC50 > 10000 nM T31204 CNB39C 10947658 Ki = 44 nM T31204 C4T8LY 11020695 Ki = 19 nM T31204 CVE8T3 11121216 Ki = 310 nM T31204 CHEV46 11148641 Ki = 681 nM T31204 CZK0E6 11150514 Ki = 3430 nM T31204 CTHA45 11151653 EC50 = 12 nM T31204 C3NH7G 11160564 EC50 = 794.33 nM T31204 C4SOG5 11163458 Ki = 380 nM T31204 C1SXY8 11171464 EC50 = 63.1 nM T31204 COG98Y 11171955 EC50 = 271 nM T31204 CLP45Z 11175045 Ki = 190 nM T31204 C6OLX8 11176570 Ki = 340 nM T31204 C4FYN6 11185858 Ki = 2350 nM T31204 CDA9Z8 11187156 Ki = 220 nM T31204 C90ZAQ 11195293 Ki = 3445 nM T31204 C52BGU 11206703 EC50 = 37 nM T31204 C5NA0Z 11209786 Ki = 209 nM T31204 C2A1PL 11221167 Ki = 74 nM T31204 CAF7T3 11222829 Ki = 5513 nM T31204 CJS0I7 11225281 Ki < 794.33 nM T31204 CZFH27 11231392 EC50 = 825 nM T31204 CXB4Q8 11233293 Ki = 29 nM T31204 CNR71Z 11235362 Ki < 1000 nM T31204 CBO29U 11236301 Ki = 125.89 nM T31204 C2JOS6 11237290 Ki = 158.49 nM T31204 C90WSG 11248705 Ki = 1584.89 nM T31204 C3XS7W 11253485 Ki = 3740 nM T31204 CWD43K 11264345 EC50 = 2511.89 nM T31204 C4S2VF 11277147 Ki = 1.8 nM T31204 CLFM61 11282335 Ki = 199.53 nM T31204 CJD16T 11288140 Ki = 3930 nM T31204 COQ7H8 11290492 Ki = 192 nM T31204 C83DSZ 11292350 Ki = 199.53 nM T31204 CM43ZJ 11300712 EC50 = 28 nM T31204 CB0UJ7 11302765 Ki = 153 nM T31204 C9BLC7 11304596 Ki = 1258.93 nM T31204 CU4L6M 11304816 IC50 = 349 nM T31204 C49LMW 11305844 Ki = 251.19 nM T31204 CLQM72 11312820 Ki = 3010 nM T31204 CU81GW 11313985 EC50 = 56 nM T31204 C1EAK6 11324968 Ki = 105 nM T31204 C46TGM 11328372 Ki < 2511.89 nM T31204 C2DVE9 11333043 EC50 > 5000 nM T31204 CV1I4W 11336079 Ki = 2099 nM T31204 CDN79K 11346775 Ki = 890 nM T31204 CHW9G0 11347858 Ki = 470 nM T31204 CU5L7F 11361103 Ki = 778 nM T31204 CF4OX6 11397149 Ki > 6309.57 nM T31204 C7IPE2 11400855 EC50 = 3092 nM T31204 C7RAB8 11414184 EC50 = 192 nM T31204 COZJ91 11416698 Ki = 196 nM T31204 CNM62W 11419526 Ki = 100 nM T31204 CIB9K8 11427139 Ki = 648 nM T31204 C3K7TG 11430311 Ki = 199.53 nM T31204 CYZC62 11437171 Ki = 84 nM T31204 CF94ZE 11447552 EC50 = 1584.89 nM T31204 CY06IJ 11448649 EC50 = 498 nM T31204 CHS2R7 11453704 Ki = 199.53 nM T31204 C1W8QL 11454107 Ki < 1000 nM T31204 CY76VX 11463745 Ki = 316.23 nM T31204 CDTI21 11465413 Ki = 251.19 nM T31204 C1QL6G 11475519 Ki = 125.89 nM T31204 CB2X1C 11483068 Ki = 248 nM T31204 CJ6GV8 11492300 Ki = 5812 nM T31204 CSP63L 11493484 Ki = 87 nM T31204 CFY18U 11499800 Ki = 191 nM T31204 CJ2O6D 11514226 Ki = 23 nM T31204 CW68BJ 11518143 IC50 = 1000 nM T31204 C9ZT5F 11536299 Ki = 2454.71 nM T31204 C5VHK0 11536843 Ki = 5.1 nM T31204 C0YZ7L 11536844 Ki = 2.7 nM T31204 CMTN14 11579853 Ki = 188 nM T31204 C90XFB 11587397 Ki = 2373 nM T31204 C5TQ3Y 11595191 Ki = 140 nM T31204 CGX8F6 11596869 Ki > 3300000 nM T31204 CZ2OG1 11608308 EC50 = 1258.93 nM T31204 CYF3M8 11609026 Ki = 48 nM T31204 C5JZ6R 11615459 Ki = 8.6 nM T31204 CN3WL4 11630147 Ki = 63 nM T31204 C9F4UK 11630623 Ki = 79 nM T31204 C9OXY8 11644842 Ki = 535 nM T31204 CVU40P 11652359 Ki = 1717 nM T31204 CM57PQ 11652452 Ki = 24 nM T31204 C1HDM5 11653679 Ki = 495.2 nM T31204 CR7WX0 11665991 Ki = 734 nM T31204 CI81RY 11666237 Ki = 478 nM T31204 CD91CP 11666595 Ki = 0.11 nM T31204 CAI7R5 11673842 Ki = 776 nM T31204 CEQ6W7 11694810 Ki = 4.3 nM T31204 CCE9H2 11695000 EC50 = 9.9 nM T31204 CU8QZ9 11701315 Ki = 280 nM T31204 CRH96P 11716185 Ki = 905 nM T31204 C53KHL 11737032 Ki = 309 nM T31204 CH0PB9 11737939 EC50 = 57 nM T31204 C05TYZ 11739217 Ki = 1300 nM T31204 C8Q4ET 11742218 Ki = 50.12 nM T31204 CPG15O 11743399 IC50 > 1000 nM T31204 CUE3K5 11749963 Ki < 10000 nM T31204 C6SKL1 11750162 Ki = 316.23 nM T31204 CK4LU1 11750342 Ki < 1000 nM T31204 CT7YB5 11753781 Ki = 199.53 nM T31204 C7KD9Z 11766873 Ki = 316.23 nM T31204 CNZV46 11774955 Ki < 1584.89 nM T31204 C4IQ8G 11775262 Ki = 199.53 nM T31204 CUT31Z 11777150 EC50 = 190 nM T31204 CQ98FK 11819486 Ki = 93.5 nM T31204 CE6J4U 11820166 Ki = 64.9 nM T31204 CAD8P9 11848624 Ki = 41 nM T31204 CM49QW 11848625 Ki = 94 nM T31204 CXLW54 11948707 Ki = 33.7 nM T31204 CQ64OY 11949706 Ki = 83 nM T31204 CP79ZF 11949710 Ki = 7.7 nM T31204 CEYG15 11949712 EC50 = 300 nM T31204 CWG8D2 11952353 Ki = 153 nM T31204 C8JQL7 11957735 IC50 = 7745 nM T31204 CR7IZ8 11983273 EC50 = 65 nM T31204 CUD9A3 12017598 Ki = 79.43 nM T31204 CM95EO 12017599 Ki = 19.95 nM T31204 CTMH07 12370465 EC50 = 85 nM T31204 CM8FI1 12370466 EC50 > 10000 nM T31204 C6I4GL 12901777 Ki = 4540 nM T31204 CCG14E 13091356 Ki = 898 nM T31204 CYN95Z 13091359 Ki = 1057 nM T31204 CPFQ95 13764011 EC50 = 1.259 nM T31204 CJ16HE 15011385 Ki = 26 nM T31204 C7VAI1 15011772 IC50 > 10000 nM T31204 C5ZK0U 15640062 EC50 = 50.12 nM T31204 CXW37K 15987265 IC50 = 3100 nM T31204 C37FIP 16047544 EC50 = 4.8 nM T31204 C6OYT5 16062136 Ki = 70 nM T31204 CBWZ28 16062137 Ki = 2500 nM T31204 CLG47H 16062139 Ki = 2250 nM T31204 C6Y3LW 16062143 Ki = 210 nM T31204 C0K1DQ 16062145 Ki = 9000 nM T31204 C9HQ7A 16062266 Ki = 2200 nM T31204 CM45DK 16062270 Ki = 220 nM T31204 C09LXV 16062651 Ki = 400 nM T31204 C8PU1B 16062781 Ki = 30 nM T31204 CCL8Z7 16062782 Ki = 1 nM T31204 C7VW3X 16062783 Ki = 4.8 nM T31204 CXQ0L4 16062784 Ki = 20 nM T31204 CKB71R 16062785 Ki = 20 nM T31204 CPS49Q 16062788 Ki = 30 nM T31204 C4AZV6 16062910 Ki = 2.5 nM T31204 CK08NX 16062911 Ki = 22 nM T31204 C4JTB1 16062912 Ki = 40 nM T31204 CQBU41 16063039 Ki = 1300 nM T31204 C16OJN 16063047 Ki = 10000 nM T31204 C51YGX 16063181 Ki = 310 nM T31204 C1SR0O 16071847 Ki = 344 nM T31204 CEWI25 16115148 Ki = 3690 nM T31204 CA15XJ 16115267 Ki = 29 nM T31204 CVL4O8 16115269 EC50 = 100 nM T31204 CA15YJ 16115271 Ki = 7 nM T31204 CU86YM 16115381 EC50 = 22 nM T31204 CCZ1E8 16115388 Ki = 235 nM T31204 C3PE9N 16115390 Ki > 10000 nM T31204 C8KMO4 16115392 EC50 = 290 nM T31204 CIN2U9 16115511 EC50 = 274 nM T31204 CJ1YO5 16115513 EC50 > 1000 nM T31204 C5RK9P 16115515 EC50 > 1000 nM T31204 C4J7OR 16115517 EC50 = 8 nM T31204 CVF2A4 16115521 Ki = 471 nM T31204 CJO13N 16115644 EC50 = 33 nM T31204 CXNA76 16115647 Ki > 10000 nM T31204 C0F5WY 16115650 Ki > 10000 nM T31204 C4IT3C 16115652 EC50 = 175 nM T31204 CWG94S 16115654 EC50 = 282 nM T31204 CZ1WJ4 16117151 Ki = 155 nM T31204 CM32ZX 16117153 Ki = 675 nM T31204 CXTB90 16117279 Ki = 1760 nM T31204 C1F2LS 16118795 Ki = 675 nM T31204 C69VDS 16118923 Ki = 33 nM T31204 C9EF6M 16215237 Ki = 100 nM T31204 CZ2IS9 16660294 Ki > 10000 nM T31204 CPT9U5 16812804 IC50 = 2.4 nM T31204 C1GR9B 17954204 EC50 = 1000 nM T31204 C3J2EH 17989823 Ki = 501.19 nM T31204 CV7T6Z 17989828 Ki < 794.33 nM T31204 CZO18R 17989871 Ki = 63.1 nM T31204 C8JEI2 17989875 Ki < 3162.28 nM T31204 C9RY6L 18005120 Ki = 39.81 nM T31204 CZ58PY 18357723 Ki = 501.19 nM T31204 C2I7CO 18357724 Ki = 251.19 nM T31204 CS90WO 18357730 Ki = 7.943 nM T31204 C82DBE 18475509 Ki = 12.59 nM T31204 C3DP7R 18475581 Ki = 630.96 nM T31204 CNP6Q1 18475610 Ki = 15.85 nM T31204 CHP8Q5 18475630 Ki = 3.981 nM T31204 C8EQN1 18475647 Ki = 50.12 nM T31204 CUZ6M7 18520432 EC50 = 31.62 nM T31204 CNAK30 18715554 EC50 = 152 nM T31204 CSIT54 18715555 EC50 = 20 nM T31204 CNFG32 18715558 EC50 = 62 nM T31204 C03DXY 18715561 EC50 = 45 nM T31204 CG2K0J 18715564 EC50 = 2.1 nM T31204 C2ST7K 18735305 EC50 = 22 nM T31204 CUC5V9 18735309 EC50 = 49 nM T31204 C9GW5T 18735313 EC50 = 6.5 nM T31204 CRLH78 18931123 Ki = 316.23 nM T31204 C42WCN 18931133 Ki = 100 nM T31204 CW7QF4 18931150 Ki = 199.53 nM T31204 CZKR20 18931163 Ki = 398.11 nM T31204 CW5GP0 18931172 Ki = 398.11 nM T31204 C7PU3Q 18931202 Ki = 50.12 nM T31204 C1INB0 18931217 Ki = 3162.28 nM T31204 CY10RA 18931344 Ki = 630.96 nM T31204 CODQ12 18931348 Ki = 125.89 nM T31204 C37ZWN 18931357 Ki = 79.43 nM T31204 C5LQX3 18931377 Ki = 199.53 nM T31204 C5T4BW 18931420 Ki = 398.11 nM T31204 CY60VR 18931422 Ki = 10 nM T31204 C1HL8Z 19356259 Ki = 316.23 nM T31204 CNJY54 20824945 Ki = 21 nM T31204 CSN4T5 20824946 Ki = 250 nM T31204 CRUI61 20824949 Ki = 960 nM T31204 CPLT36 21044391 Ki = 1139 nM T31204 C6JSC0 21044398 Ki = 835 nM T31204 CWHT46 21302483 Ki = 15 nM T31204 C3T5HF 21509921 Ki = 87 nM T31204 CFN81Q 21527771 Ki = 1622 nM T31204 CH59WN 21533446 Ki = 790 nM T31204 CQO1R3 21786603 Ki = 116 nM T31204 CT7XG9 21830793 Ki = 73.6 nM T31204 CO32YX 22254068 Ki = 245 nM T31204 CQMS26 22292784 EC50 = 501.19 nM T31204 CC6AJ0 22368315 EC50 = 400 nM T31204 C5IE1F 22619858 Ki = 125.89 nM T31204 C81XUE 23027035 IC50 = 120 nM T31204 CR5H1I 23027211 IC50 = 130 nM T31204 CC2L1B 23027245 IC50 = 170 nM T31204 CG9M4Y 23027411 IC50 = 300 nM T31204 CC6R2O 23027527 IC50 = 300 nM T31204 C5BUL7 23151712 Ki = 18 nM T31204 C3IF7P 23151734 Ki = 0.4 nM T31204 C0NI3J 23290944 Ki = 327 nM T31204 C1RIA7 23395431 EC50 = 794.33 nM T31204 CA6QL5 23462894 Ki = 1000 nM T31204 C0U2TC 23467920 EC50 > 10000 nM T31204 CR1M4E 23652278 EC50 = 1258.93 nM T31204 C67YVI 24740863 Ki = 74 nM T31204 CD7CV6 24771120 Ki = 130 nM T31204 CGX8K2 24773648 EC50 < 10000 nM T31204 CSCJ40 24773649 EC50 = 39.81 nM T31204 C6T5XP 24773650 EC50 = 199.53 nM T31204 CLR9M6 24773651 EC50 = 39.81 nM T31204 CMA8Q6 24773728 EC50 = 630.96 nM T31204 C4O2YA 24773809 EC50 = 501.19 nM T31204 C7IT2S 24773814 EC50 = 251.19 nM T31204 C2U8IH 24773816 EC50 = 251.19 nM T31204 CTK36B 24773894 EC50 < 10000 nM T31204 CG1V5R 24773895 EC50 = 398.11 nM T31204 C9WV5A 24773897 EC50 < 10000 nM T31204 C6IF2A 24773900 EC50 = 780 nM T31204 CNOE28 24773901 EC50 > 5000 nM T31204 C8R9DY 24773978 EC50 < 10000 nM T31204 CF2U4K 24773979 EC50 = 3981.07 nM T31204 CJN09A 24826786 Ki = 213 nM T31204 C3PQB2 24826787 Ki = 47 nM T31204 CRKE01 24826788 Ki = 8 nM T31204 C6BM3J 24826790 Ki = 13 nM T31204 CF9VK5 24826867 Ki = 2 nM T31204 CJ7Q4O 24826868 EC50 = 9 nM T31204 CT8R9F 24826869 EC50 = 28 nM T31204 C8W9FT 24826870 Ki = 227 nM T31204 CSDP50 24826871 Ki = 78 nM T31204 CGQZ94 24826957 Ki = 17 nM T31204 C5DZ6K 24826963 Ki = 21 nM T31204 CDC91N 24839550 Ki = 61.66 nM T31204 CY21RE 24841480 Ki = 100 nM T31204 CBA17N 24849050 EC50 = 62 nM T31204 C3HK0J 24865725 Ki = 1995.26 nM T31204 C0O6FX 24865727 Ki > 1000 nM T31204 C0KFD3 24884789 Ki < 10000 nM T31204 C2NT1L 24887284 Ki = 1584.89 nM T31204 C2J0BI 24887285 Ki < 1584.89 nM T31204 CB41AM 24887289 Ki < 1584.89 nM T31204 CC2IJ9 24887290 Ki = 501.19 nM T31204 CXJ90O 24887291 Ki < 5011.87 nM T31204 CTDX79 24887517 Ki = 1995.26 nM T31204 C6L7KS 24887518 Ki = 630.96 nM T31204 CPY96D 24887519 Ki < 1584.89 nM T31204 C90ACW 24887525 Ki = 1000 nM T31204 CR31BN 24887527 Ki = 501.19 nM T31204 C2NVO1 24887761 Ki < 1584.89 nM T31204 C17OXP 24887768 Ki < 1584.89 nM T31204 C24NPA 24887966 Ki < 1584.89 nM T31204 C04UDV 24887967 Ki < 794.33 nM T31204 CHA0N5 24887968 Ki < 1000 nM T31204 CX04AI 24887970 Ki < 794.33 nM T31204 C0DX5I 24888180 Ki = 630.96 nM T31204 CO74UR 24888181 Ki = 1000 nM T31204 CGLH34 24888182 Ki < 5011.87 nM T31204 C6R9EH 24888183 Ki = 1584.89 nM T31204 CZX93A 24888184 Ki < 1000 nM T31204 C1GR0V 24888185 Ki < 630.96 nM T31204 CI53SE 24893978 Ki = 140 nM T31204 C3C0KP 24894134 EC50 > 50000 nM T31204 CW4X0E 24962988 EC50 > 10000 nM T31204 C1PKF0 25056080 Ki = 7943.28 nM T31204 CTI38U 25060119 Ki = 662 nM T31204 CYJ5G1 25067564 Ki = 274 nM T31204 C4B0FU 25070577 IC50 = 110 nM T31204 COG5H7 25070581 EC50 = 164 nM T31204 CBY3O2 25070582 EC50 > 10000 nM T31204 CZOW25 25070907 EC50 = 183 nM T31204 C3H2FL 25070909 EC50 > 10000 nM T31204 CK0FZ5 25070911 EC50 = 247 nM T31204 CO48CT 25071230 EC50 > 10000 nM T31204 C9SZG1 25084025 EC50 = 141 nM T31204 CR17NY 25110703 Ki = 398.11 nM T31204 CNS84K 25117676 Ki = 423 nM T31204 C4WV0K 25117677 Ki = 583 nM T31204 CL19XF 25117679 Ki = 185 nM T31204 CWFY19 25117680 Ki = 191 nM T31204 CSW9K6 25117681 Ki > 3300 nM T31204 CA1EJ2 25120700 Ki = 164 nM T31204 C1PG8Z 25122651 Ki = 100 nM T31204 CD3R5U 25122652 Ki = 493 nM T31204 CK58IM 25122653 Ki = 78 nM T31204 CA12QG 25122654 Ki = 442 nM T31204 C3M0EY 25123011 Ki = 1362 nM T31204 CZX2R0 25123012 Ki > 10000 nM T31204 CNV98C 25123013 Ki = 97.9 nM T31204 C3N6SM 25123014 Ki = 21 nM T31204 CGH08V 25164128 Ki = 794.33 nM T31204 C5C7GH 25184832 Ki = 794.33 nM T31204 CN06PX 25209050 Ki = 64.57 nM T31204 CR1K8B 25209356 Ki = 1698.24 nM T31204 CLKT16 25209357 Ki > 4786.3 nM T31204 CDF83Q 25209705 Ki = 912.01 nM T31204 CJ1Z9H 25216680 Ki > 10000 nM T31204 C1T3LR 25218143 Ki > 10000 nM T31204 CPI03N 25218397 Ki > 10000 nM T31204 CL1R3Q 25218401 Ki > 10000 nM T31204 CM2T9Y 25263297 Ki = 155 nM T31204 CFJM71 25263302 Ki = 174 nM T31204 CH67OW 26694436 IC50 = 230 nM T31204 C4MRQ0 27842480 Ki = 674 nM T31204 C1D2LR 29943048 Ki = 3.2 nM T31204 CA58DL 41305446 Ki = 569 nM T31204 CTI9S6 42601404 EC50 > 9940 nM T31204 CQR2J6 42601405 EC50 = 18 nM T31204 CJ3NP5 42636941 IC50 = 281.84 nM T31204 C0AI7N 43229249 Ki = 273 nM T31204 C16UIM 44138039 IC50 = 0.2 nM T31204 CV4TD7 44155107 IC50 = 411 nM T31204 C6TND7 44155109 IC50 = 161 nM T31204 CXM4K7 44156628 Ki = 464 nM T31204 CY41DQ 44156752 Ki = 188 nM T31204 C73FZD 44156754 Ki = 153 nM T31204 CPE0L5 44156863 IC50 = 118 nM T31204 C2AV1K 44190762 IC50 = 1140 nM T31204 CQ8NV3 44214723 Ki = 25.12 nM T31204 CSVN47 44214724 Ki = 10 nM T31204 CJ8F5Y 44215629 Ki = 65 nM T31204 CRNL71 44225654 EC50 > 9940 nM T31204 C09VPJ 44243470 Ki = 3160 nM T31204 C1DX4N 44269058 Ki = 2.2 nM T31204 C7Z4RE 44275982 Ki > 10000 nM T31204 CU35RG 44276349 Ki = 6470 nM T31204 CG62JB 44298021 Ki = 199.53 nM T31204 CV5YP3 44298022 Ki = 100 nM T31204 CY1B3H 44298079 Ki = 1995.26 nM T31204 CCU89I 44298080 Ki = 6.31 nM T31204 C9TS2N 44298082 Ki = 15.85 nM T31204 CY0VX7 44298086 Ki = 39.81 nM T31204 CSIC31 44298091 Ki = 630.96 nM T31204 CZ7BV3 44298092 Ki = 100 nM T31204 CO06KG 44298100 Ki = 501.19 nM T31204 C1AF0K 44298108 Ki = 100 nM T31204 C9AVQ8 44298118 Ki = 19.95 nM T31204 C6Z0QR 44298120 Ki = 251.19 nM T31204 C41MRW 44298121 Ki = 25.12 nM T31204 CP0D3F 44298126 Ki = 2511.89 nM T31204 C3KUI9 44298129 Ki = 5011.87 nM T31204 CH2UE9 44298138 Ki = 199.53 nM T31204 CPL7S5 44298140 Ki = 398.11 nM T31204 CJ3H6P 44298142 Ki = 794.33 nM T31204 C1SBI3 44298147 Ki > 10000 nM T31204 CI9S7T 44298151 Ki = 1000 nM T31204 CUQ5J7 44298157 Ki > 1995.26 nM T31204 CV14AJ 44298158 Ki = 1000 nM T31204 CG46JN 44298163 Ki = 12.59 nM T31204 CE8C1H 44298172 Ki = 12.59 nM T31204 CS6XN2 44298173 Ki = 31.62 nM T31204 CO9YU5 44298175 Ki = 50.12 nM T31204 C93TDS 44298176 Ki = 7.943 nM T31204 CIP20E 44298182 Ki = 630.96 nM T31204 C5EDF3 44298186 Ki = 251.19 nM T31204 C71ZLS 44298192 Ki = 316.23 nM T31204 C0IC9T 44298193 Ki = 1995.26 nM T31204 CX64BM 44298208 Ki = 79.43 nM T31204 CF1K0H 44298209 Ki = 63.1 nM T31204 C7L1FM 44298225 Ki = 63.1 nM T31204 C3NK6M 44298226 Ki = 158.49 nM T31204 CU0FL2 44298229 Ki = 19.95 nM T31204 CE1Y5J 44298230 Ki = 100 nM T31204 C0N3KH 44298234 Ki = 39.81 nM T31204 C9YRS1 44298236 Ki = 31.62 nM T31204 C14RQX 44298243 Ki = 125.89 nM T31204 CWC4O2 44298244 Ki = 63.1 nM T31204 C58LBP 44298246 Ki = 12.59 nM T31204 CX2WP8 44298249 Ki = 25.12 nM T31204 C2Q5ZP 44298254 Ki = 125.89 nM T31204 CT1JY4 44299663 Ki = 79.43 nM T31204 CP0C2G 44315697 EC50 = 31 nM T31204 CF40WU 44315993 EC50 = 10 nM T31204 C1GQT9 44316017 EC50 = 7.3 nM T31204 CS25VN 44316027 EC50 = 72 nM T31204 CEA13Y 44323840 Ki = 251.19 nM T31204 CPB89X 44323908 Ki < 10000 nM T31204 C3MXG7 44324011 Ki = 125.89 nM T31204 CGOY42 44324142 Ki = 6.31 nM T31204 CPWJ26 44343212 Ki = 3981.07 nM T31204 CUXH48 44352308 Ki = 676 nM T31204 CX38YF 44364163 Ki = 5.7 nM T31204 C6M0VT 44364215 Ki = 38.1 nM T31204 C8DVZ6 44364514 Ki = 58.3 nM T31204 C4MLR3 44389645 EC50 = 220 nM T31204 CUR07Z 44389646 EC50 = 30 nM T31204 C50AJV 44393215 IC50 = 400 nM T31204 C90NSU 44393396 IC50 = 201 nM T31204 C4B0OI 44397588 Ki = 1258.93 nM T31204 C5FP0R 44397589 Ki = 1995.26 nM T31204 CE3G8U 44397670 Ki = 1000 nM T31204 CQR59X 44397731 Ki = 90 nM T31204 C8VJ5H 44397752 Ki = 67 nM T31204 C8EQU9 44397832 Ki = 11 nM T31204 CYDA14 44397846 Ki = 59 nM T31204 C0FUY7 44397929 Ki = 10 nM T31204 CUVA58 44404608 Ki = 1258.93 nM T31204 C53KTE 44404616 Ki > 6309.57 nM T31204 C4XIR6 44404619 Ki > 7943.28 nM T31204 CW1BK6 44404623 Ki > 5011.87 nM T31204 CHG15M 44404887 Ki = 170 nM T31204 CL9GC3 44404895 Ki = 5566 nM T31204 CW20SO 44407327 EC50 = 462 nM T31204 COY19S 44407335 EC50 = 128 nM T31204 CW57QU 44407337 EC50 = 91 nM T31204 C6Z5PB 44407398 EC50 = 27 nM T31204 C2Q5MJ 44407440 EC50 = 128 nM T31204 CR1D5Y 44407453 EC50 = 44 nM T31204 CL94HP 44407460 EC50 = 97 nM T31204 COH25L 44409031 Ki = 48 nM T31204 C4TZ7J 44409032 Ki = 217 nM T31204 C6I4CY 44409095 Ki = 440 nM T31204 CWX62Y 44409096 Ki = 77 nM T31204 CM6ZY0 44409097 Ki = 68 nM T31204 CJ8UB2 44409101 Ki = 379 nM T31204 C5K2ZG 44409124 Ki = 1820 nM T31204 CG87PW 44409290 EC50 = 23 nM T31204 CI69ML 44409316 Ki = 81 nM T31204 CMP47G 44409317 Ki = 166 nM T31204 CIPR62 44409327 Ki = 295 nM T31204 CPDN92 44409332 Ki = 1306 nM T31204 CQLM69 44412150 EC50 = 320 nM T31204 C0VIZ4 44412388 EC50 = 48 nM T31204 CZV87X 44412389 EC50 = 151 nM T31204 CA7CM1 44412403 EC50 = 59 nM T31204 C7R5WO 44412404 EC50 = 108 nM T31204 CA1SO2 44412405 EC50 = 187 nM T31204 C95IMP 44414051 Ki = 501.19 nM T31204 C9W3KV 44414057 Ki < 1995.26 nM T31204 C2JIS7 44414070 Ki = 199.53 nM T31204 CKM83W 44414105 Ki = 316.23 nM T31204 C1MQU7 44414127 Ki < 1000 nM T31204 C84CDF 44414132 Ki < 1000 nM T31204 CX10RT 44414133 Ki < 1000 nM T31204 C5HPJ4 44414150 Ki < 1584.89 nM T31204 C6ZTK1 44414164 Ki < 1584.89 nM T31204 CA4MG3 44414179 Ki < 1584.89 nM T31204 CU7G6H 44414192 Ki < 1995.26 nM T31204 C5EO1B 44414209 Ki = 1258.93 nM T31204 C9WJD2 44414217 Ki = 1584.89 nM T31204 CQ1H9S 44414233 Ki < 10000 nM T31204 CQ13GM 44414244 Ki < 1584.89 nM T31204 COY3V0 44414251 Ki = 199.53 nM T31204 CQ6K7F 44414267 Ki < 1000 nM T31204 CKG9P2 44414300 Ki < 3162.28 nM T31204 C39GJK 44416247 IC50 = 115 nM T31204 C0WTV8 44416259 IC50 = 26 nM T31204 C0YV1G 44416260 IC50 = 32 nM T31204 CF0C1M 44416290 IC50 = 16 nM T31204 CV1JC2 44416309 IC50 = 21 nM T31204 C6T3AF 44416351 IC50 = 5000 nM T31204 CK9R1S 44420682 EC50 = 417 nM T31204 C6PBE9 44420683 Ki = 3190 nM T31204 C7KBP0 44430566 Ki < 6309.57 nM T31204 CBP57S 44430955 Ki < 794.33 nM T31204 CIZ54L 44430956 Ki < 199.53 nM T31204 C1FHD3 44430958 Ki < 7943.28 nM T31204 CX0O2S 44430974 Ki < 3162.28 nM T31204 CQFV73 44430976 Ki = 125.89 nM T31204 CG0CH7 44430979 Ki = 125.89 nM T31204 C14ZCW 44430984 Ki < 1000 nM T31204 CZ3RM2 44435219 Ki = 2000 nM T31204 CKZF16 44439165 Ki < 1000 nM T31204 CA4HZ3 44439167 Ki = 3162.28 nM T31204 CZL95J 44451390 Ki = 210 nM T31204 CL14SE 44451393 Ki = 84 nM T31204 C32AJU 44451422 Ki = 410 nM T31204 CT5JO6 44451429 Ki = 300 nM T31204 C78NHG 44453103 Ki = 70 nM T31204 C4L6TY 44453652 Ki = 270 nM T31204 CVN1O4 44453877 Ki = 1000 nM T31204 CZL97F 44455426 Ki = 299 nM T31204 C12XGE 44456400 Ki = 562.34 nM T31204 CXY7T9 44476436 IC50 = 6160 nM T31204 C1H8NX 44516817 Ki = 1040 nM T31204 C3D4HR 44537940 Ki = 141 nM T31204 CJ7U3K 44554227 Ki = 96 nM T31204 CM0I1P 44554393 Ki = 281 nM T31204 CNHA47 44554395 Ki = 87 nM T31204 CUQ0J7 44555369 EC50 > 10000 nM T31204 C7K4CG 44565605 IC50 = 710 nM T31204 CI59JV 44565606 IC50 = 4 nM T31204 CH6K4V 44565607 IC50 = 6 nM T31204 CQH8Z1 44565608 IC50 = 0.6 nM T31204 CYV4D1 44565633 IC50 > 1300 nM T31204 CQ23DW 44565634 IC50 = 340 nM T31204 CO13NS 44565635 IC50 = 15 nM T31204 CWP6Y2 44565636 IC50 = 120 nM T31204 C5A2BT 44565637 IC50 = 22 nM T31204 CF73ZH 44565638 IC50 = 840 nM T31204 CL7A1J 44565639 IC50 = 7300 nM T31204 CLTN16 44565640 IC50 = 6900 nM T31204 CTFL86 44565641 IC50 = 150 nM T31204 CSG4M5 44565805 IC50 = 31 nM T31204 C9DZ1A 44565806 IC50 = 48 nM T31204 CA28BI 44565807 IC50 = 2300 nM T31204 C9ZB2S 44565808 IC50 = 3200 nM T31204 C4QB2T 44565824 IC50 = 95 nM T31204 CXAV89 44565825 IC50 > 24000 nM T31204 CN63MU 44565826 IC50 = 610 nM T31204 C78JQI 44565827 IC50 = 12 nM T31204 CVI53P 44565828 IC50 = 10000 nM T31204 CS1H4L 44565829 IC50 = 1500 nM T31204 C56TGX 44565830 IC50 = 2.4 nM T31204 C72MEU 44565831 IC50 = 0.4 nM T31204 C6LAO0 44565846 IC50 = 2.3 nM T31204 CK9D7P 44565847 IC50 = 0.3 nM T31204 CV5WK9 44565848 IC50 = 6.5 nM T31204 C7J8IR 44565849 IC50 = 1100 nM T31204 CF46TU 44565850 IC50 = 1.1 nM T31204 CVA67X 44568347 Ki = 630 nM T31204 CGFE18 44572164 EC50 = 459 nM T31204 CWG32I 44572166 Ki = 16 nM T31204 C9B3LM 44572168 EC50 = 14 nM T31204 CYS32A 44572170 EC50 = 83 nM T31204 CX93AL 44572172 EC50 = 4.9 nM T31204 C9PGC5 44572174 EC50 = 7 nM T31204 C07DQB 44572176 EC50 = 116 nM T31204 CS26GU 44572178 EC50 = 8.4 nM T31204 CJA7V6 44572180 EC50 = 12 nM T31204 CYOJ47 44572207 EC50 = 116 nM T31204 CV52SZ 44572252 EC50 > 1000 nM T31204 CB81WN 44572254 EC50 > 1000 nM T31204 C69CUA 44572304 EC50 > 1000 nM T31204 CXU7Z8 44572367 EC50 = 204 nM T31204 C6GIR9 44572369 EC50 = 185 nM T31204 CY5Q8G 44572371 EC50 = 1739 nM T31204 C7WJS5 44572657 EC50 = 37 nM T31204 COK9N1 44572698 EC50 = 510 nM T31204 C9QJB3 44572747 EC50 = 69 nM T31204 C6S2DJ 44572749 EC50 = 32 nM T31204 C97VKX 44572751 EC50 = 13 nM T31204 C2AQR8 44572753 EC50 = 224 nM T31204 C2RV0K 44572755 EC50 = 53 nM T31204 CKIC03 44572757 EC50 = 350 nM T31204 CQU5B9 44572759 EC50 = 199 nM T31204 CYTA39 44572761 EC50 = 492 nM T31204 C6CGB5 44572798 EC50 = 3.6 nM T31204 C20GHO 44572800 EC50 = 59 nM T31204 CJ1VI8 44572802 EC50 = 65 nM T31204 CLV5I8 44572804 EC50 = 77 nM T31204 C43IDZ 44572806 EC50 = 75 nM T31204 CT64CF 44572808 EC50 = 5.5 nM T31204 CU25XD 44572810 EC50 = 21 nM T31204 CS7KZ5 44572812 EC50 = 404 nM T31204 C6QFY7 44573002 EC50 = 2737 nM T31204 CP16NR 44573004 EC50 = 37 nM T31204 C9MXB5 44573006 EC50 > 1000 nM T31204 CQ70OY 44573012 EC50 = 366 nM T31204 CE95AX 44573014 EC50 = 415 nM T31204 CEC7J9 44573016 EC50 = 3342 nM T31204 CUB38Y 44573018 EC50 = 28 nM T31204 CI3V4D 44573153 EC50 = 478 nM T31204 CX1N8H 44573154 EC50 = 802 nM T31204 C7C5ZW 44573155 EC50 = 103 nM T31204 C3L0BU 44573156 EC50 = 125 nM T31204 CD9V7Q 44573157 EC50 = 478 nM T31204 CZM8O6 44573159 EC50 > 9940 nM T31204 CVSJ62 44573160 EC50 > 9940 nM T31204 CF0A2J 44573161 EC50 > 9940 nM T31204 C13LFI 44573162 EC50 > 9940 nM T31204 CB60NZ 44573165 EC50 > 9940 nM T31204 C0F5DM 44573216 EC50 = 197 nM T31204 C6X3QF 44573217 EC50 = 69 nM T31204 CF9X3C 44573218 EC50 = 75 nM T31204 CUC43W 44573219 EC50 > 9940 nM T31204 C4I8AJ 44573220 EC50 = 17 nM T31204 CXDU28 44573221 EC50 = 357 nM T31204 C2HS3V 44573222 EC50 = 34 nM T31204 C7HZJ6 44573224 EC50 > 9940 nM T31204 C46QXT 44573225 EC50 > 9940 nM T31204 CKSA47 44573226 EC50 > 9940 nM T31204 CD62CX 44573227 EC50 > 9940 nM T31204 CDH04E 44573229 EC50 = 18 nM T31204 CAF64P 44573230 EC50 = 33 nM T31204 CPK71S 44573231 EC50 = 15 nM T31204 C5TKU6 44579715 Ki = 2390 nM T31204 C5NS6H 44581972 Ki = 154.88 nM T31204 CK8Z1P 44581973 Ki = 30.2 nM T31204 C3UQ9Z 44581974 Ki = 97.72 nM T31204 CRCH48 44582675 Ki = 320 nM T31204 CEJ4R8 44582676 Ki = 960 nM T31204 CZGP86 44582677 Ki = 1844 nM T31204 C5QB4K 44582678 Ki = 466 nM T31204 C01RCI 44582705 Ki = 559 nM T31204 CXL25V 44582706 Ki = 2751 nM T31204 C8MR1X 44582707 Ki = 1052 nM T31204 C4IT1N 44582708 Ki = 1972 nM T31204 CB0S4Z 44592109 IC50 = 52.48 nM T31204 C43LPI 44622848 EC50 = 358 nM T31204 CU3LE6 44626329 Ki = 680 nM T31204 CZHP95 44626357 EC50 > 2610 nM T31204 CPEY83 45378934 Ki = 455 nM T31204 CU36SC 45378935 Ki > 3300 nM T31204 CHNI56 45378936 Ki = 260 nM T31204 C0CHF4 45482789 IC50 = 2470 nM T31204 CG8JT5 45484649 EC50 > 10000 nM T31204 CK32TH 45484650 EC50 > 10000 nM T31204 C0QP1B 45484661 EC50 = 94 nM T31204 C7JR1B 45484662 EC50 = 81 nM T31204 C2YM6L 45484673 EC50 = 267 nM T31204 C5MXW4 45484682 EC50 = 473 nM T31204 CG7SD9 45484686 EC50 > 10000 nM T31204 CB53ZY 45484687 EC50 = 142 nM T31204 CR14VO 45484700 EC50 = 84 nM T31204 CZU53K 45484701 EC50 > 10000 nM T31204 CL16EH 45484708 EC50 > 10000 nM T31204 CIF58O 45484726 EC50 > 10000 nM T31204 CJM13Y 45484727 EC50 > 10000 nM T31204 C9K7HM 45484741 EC50 > 10000 nM T31204 CQM85L 45484742 EC50 = 353 nM T31204 CGLF37 45484995 IC50 = 320 nM T31204 CGOS24 45485061 IC50 > 10000 nM T31204 CLX9C8 45485062 IC50 = 31 nM T31204 C9NK6I 45485725 EC50 = 506 nM T31204 CVK8W9 45485742 EC50 = 187 nM T31204 CD80KX 45485751 EC50 > 10000 nM T31204 CNX23T 45485779 EC50 > 10000 nM T31204 CO6Z1P 45485781 EC50 > 10000 nM T31204 CQMJ83 45486820 Ki = 165 nM T31204 CJN7X0 45486824 Ki = 6 nM T31204 C9BSL5 45486891 Ki = 400 nM T31204 C4H7OT 45486902 Ki = 110 nM T31204 CIV92F 46214153 Ki = 74 nM T31204 CF6BQ7 46228422 EC50 = 748 nM T31204 C23DJK 46228430 EC50 = 998 nM T31204 CTES15 46228437 EC50 = 397 nM T31204 CZ5MW9 46228438 EC50 = 187 nM T31204 C98NCA 46230046 Ki = 137 nM T31204 C3LMQ6 46230047 Ki = 61 nM T31204 C0D4IZ 46230048 Ki = 2395 nM T31204 C6UMX7 46230049 Ki = 18 nM T31204 C87JZL 46230094 Ki = 72 nM T31204 CINK61 46230095 Ki = 13 nM T31204 C6N7AF 46230096 Ki > 10000 nM T31204 C7WO5P 46230097 Ki = 67 nM T31204 CP0T5Y 46230098 Ki = 10 nM T31204 CPA62G 46230099 Ki = 23 nM T31204 CWQD49 46230100 Ki = 41 nM T31204 CA4HD5 46830134 IC50 = 127 nM T31204 C6K0MF 46830177 Ki = 3940 nM T31204 C0HCI4 46867519 Ki = 169 nM T31204 C6KBJ2 46882133 Ki > 10000 nM T31204 CNL16U 46882180 Ki > 10000 nM T31204 CI96SR 46884034 Ki = 3500 nM T31204 C6EL4F 46884036 Ki > 10000 nM T31204 CEUD30 46884098 Ki = 4120 nM T31204 CNET68 46884100 Ki = 2400 nM T31204 C8Y0IG 46884101 Ki = 1720 nM T31204 C5BFY9 46884102 Ki = 1670 nM T31204 C1ORQ0 46884137 EC50 > 10000 nM T31204 C3BW2P 46884138 EC50 = 4027 nM T31204 CA75HK 46914485 Ki = 9.7 nM T31204 C9D7UW 46914486 Ki = 28 nM T31204 COB4R0 46914487 Ki = 15 nM T31204 C4JZR8 46914620 Ki = 72 nM T31204 C4JIP7 46914621 Ki = 302 nM T31204 CZ5TS4 46914771 Ki = 262 nM T31204 C1LY6Z 46914772 Ki = 57 nM T31204 C3XE4P 46914773 Ki = 244 nM T31204 C2E6UX 46914774 Ki = 116 nM T31204 CT36AF 46914775 Ki = 259 nM T31204 CW74CK 46914776 Ki = 655 nM T31204 CLC27S 46914777 Ki = 184 nM T31204 CAT12G 46914926 Ki = 188 nM T31204 CE6SQ2 46914927 Ki = 232 nM T31204 CG7WR2 46933089 Ki = 1584.89 nM T31204 CW4N5K 46933090 Ki = 25.12 nM T31204 CZO5F8 46933091 Ki = 100 nM T31204 CX7R3H 46933845 EC50 = 3.981 nM T31204 CV8A5L 46937339 EC50 = 289 nM T31204 C0H1AC 46945446 Ki = 8357 nM T31204 C2LZJ0 49783209 Ki = 66 nM T31204 C57SMG 49783415 Ki = 2861 nM T31204 C0TG6I 49783419 Ki = 168 nM T31204 CD53RT 49833882 Ki = 25.12 nM T31204 C5Y4DE 49833883 Ki = 15.85 nM T31204 CGT73Y 49833884 Ki = 63.1 nM T31204 CKL16R 49833886 Ki = 158.49 nM T31204 C3KSZ8 49834050 Ki > 794.33 nM T31204 C9QS2K 49834051 Ki > 794.33 nM T31204 CF4SX0 49834052 Ki > 794.33 nM T31204 C52GPW 49834053 Ki = 316.23 nM T31204 CO20JE 49836187 Ki > 1995.26 nM T31204 CG0LF8 49836189 Ki > 1995.26 nM T31204 C0UI3V 49836294 Ki = 1258.93 nM T31204 CT7CV0 49836295 Ki > 1995.26 nM T31204 CVG9X5 49836296 Ki > 1995.26 nM T31204 C5E2ZK 49836298 Ki > 1995.26 nM T31204 CYJW87 49836299 Ki = 158.49 nM T31204 C0MS8L 49836300 Ki = 3.162 nM T31204 CR40BA 49836386 IC50 > 10000 nM T31204 CKS86Q 49836409 Ki = 251.19 nM T31204 C8E6WA 49836410 Ki > 1995.26 nM T31204 CE0PN6 49836411 Ki = 1000 nM T31204 C0I4EC 49836412 Ki = 1258.93 nM T31204 C5HU1D 49836413 Ki > 1995.26 nM T31204 C1UGC7 49836414 Ki > 1995.26 nM T31204 C0M5XC 49836496 IC50 > 10000 nM T31204 C5ZV2Y 49836522 Ki = 1258.93 nM T31204 C1JTH9 49836524 Ki = 100 nM T31204 C90XTY 49836525 Ki = 10 nM T31204 CK5QW9 49836526 Ki = 1000 nM T31204 C8RL7C 49836527 Ki > 1995.26 nM T31204 CNM9X8 49836528 Ki = 398.11 nM T31204 COK75S 49836633 Ki = 79.43 nM T31204 CZ6F7L 49836634 Ki = 39.81 nM T31204 CRM28S 49836635 Ki = 251.19 nM T31204 CA6QB8 49836636 Ki > 1995.26 nM T31204 CB81YG 49836637 Ki > 1995.26 nM T31204 CX43UC 49836639 Ki = 1584.89 nM T31204 CEBP01 49836737 Ki > 1995.26 nM T31204 CCMJ40 49836738 Ki > 1995.26 nM T31204 C3OK9Y 49836740 Ki > 1995.26 nM T31204 C26NFU 49836741 Ki > 1995.26 nM T31204 C6YM8W 49836842 Ki > 1995.26 nM T31204 C4R2YS 49850567 Ki = 794.33 nM T31204 C07JTU 49850570 Ki = 398.11 nM T31204 CK68QR 49850672 Ki = 199.53 nM T31204 CN5XR1 49850772 Ki = 79.43 nM T31204 CR4EZ0 49850870 Ki = 398.11 nM T31204 C5K4EC 49850872 Ki = 158.49 nM T31204 C8AW0R 49850874 Ki = 125.89 nM T31204 C6OQV2 49862237 Ki = 180 nM T31204 CDHY90 49864027 Ki = 96 nM T31204 CZ2SA8 49864841 Ki = 316.23 nM T31204 C2OCZ3 49864885 Ki > 1995.26 nM T31204 CS4Z8A 49864886 Ki = 630.96 nM T31204 CN8XT2 49865829 Ki = 223 nM T31204 C1FMH5 49865830 Ki = 569 nM T31204 C1CX5F 49865831 Ki = 384 nM T31204 C8RYW1 49865832 Ki = 489 nM T31204 C5ED3T 49865833 Ki = 1606 nM T31204 CAU15V 49865885 Ki > 10000 nM T31204 CLS0F3 49865886 Ki = 6596 nM T31204 CIG69Z 49865887 Ki = 1773 nM T31204 C5YEG8 49865888 Ki > 10000 nM T31204 CXP91V 49865889 Ki > 10000 nM T31204 C98TVK 49865890 Ki = 3999 nM T31204 C2RY0J 50878551 EC50 = 5.495 nM T31204 C1W6TV 50898777 Ki = 316.23 nM T31204 CXMZ73 50898778 Ki > 10000 nM T31204 CW9SV5 50942111 EC50 = 503 nM T31204 CE4KP1 51050257 Ki > 10000 nM T31204 CI90RZ 51094588 EC50 > 10000 nM T31204 C7OZN4 52944115 Ki = 15.85 nM T31204 CNQF49 52945978 Ki > 1995.26 nM T31204 C0AY5O 53317923 EC50 = 215 nM T31204 CC0T6E 53317924 EC50 = 1184 nM T31204 C1T3AI 53317925 EC50 = 73 nM T31204 C3CT4H 53320653 EC50 = 842 nM T31204 C40VGZ 53321865 EC50 = 706 nM T31204 C7LE3I 53321947 EC50 = 2242 nM T31204 CC3DB8 53321948 EC50 = 13 nM T31204 CUNP37 53323196 EC50 = 1478 nM T31204 C32YWL 53324045 Ki = 374 nM T31204 CJ9I7U 53324165 EC50 = 602 nM T31204 CQVR02 53324327 EC50 = 1158 nM T31204 CR4W9L 53324553 Ki = 6983 nM T31204 CN8X4Z 53324629 EC50 = 2848 nM T31204 C8DL1N 53324630 EC50 = 94 nM T31204 CRQF15 53325242 Ki = 423 nM T31204 CB37XF 53325861 Ki = 6086 nM T31204 C2ZFP8 53325935 EC50 = 94 nM T31204 CNE6Q8 53325936 EC50 = 218 nM T31204 C8VUJ6 53325937 EC50 = 163 nM T31204 CMB09H 53325938 EC50 = 379 nM T31204 C7J8ZY 53327611 IC50 = 1500 nM T31204 CG24AT 53381002 Ki = 88 nM T31204 CMOZ61 53475319 Ki = 762 nM T31204 CQG92V 53483975 Ki = 155 nM T31204 C6WR0E 54580776 EC50 = 178 nM T31204 C74EGT 54581791 EC50 = 60 nM T31204 C3GCR2 54583742 EC50 = 220 nM T31204 CV1IF6 54583743 EC50 = 30 nM T31204 CIC92Q 54584721 EC50 = 610 nM T31204 C46WCJ 54585653 EC50 = 160 nM T31204 C96UOS 54587668 EC50 = 1200 nM T31204 CTE1V3 54587669 EC50 = 410 nM T31204 CJRG27 54761054 Ki = 1900 nM T31204 C8YLU4 54764239 Ki = 7890 nM T31204 C01CPY 54764240 Ki = 5240 nM T31204 C42RWP 54764241 Ki = 5380 nM T31204 CA54LD 56597090 Ki = 0.6 nM T31204 C6W1RA 56649648 Ki = 99 nM T31204 C2SW7J 56649649 Ki = 79 nM T31204 CQTR49 56649650 Ki = 88 nM T31204 CY7L0C 56658155 Ki = 120 nM T31204 CFD2M9 56658156 Ki = 628 nM T31204 CD51XT 56658157 Ki = 275 nM T31204 C8RWM0 56661666 Ki = 343 nM T31204 CH37LU 56663451 IC50 > 10000 nM T31204 CSH86Y 56665074 Ki = 290 nM T31204 C6LV0H 56665075 Ki = 463 nM T31204 CY6D5E 56675412 Ki = 147 nM T31204 C4B2UC 56675413 Ki = 332 nM T31204 CEV53O 56678761 Ki = 243 nM T31204 C8H1LP 56682068 Ki = 352 nM T31204 CJKO58 56852956 Ki = 46.77 nM T31204 C1TC7Q 56963799 Ki > 10000 nM T31204 C6HBG0 57396813 Ki = 6200 nM T31204 CX0B5M 57403525 Ki = 723 nM T31204 C59YAC 57495353 IC50 = 7700 nM T31204 CDG58R 57799306 EC50 = 31 nM T31204 CS6BM2 57799321 Ki = 6244 nM T31204 CUYA69 57799324 Ki = 4 nM T31204 CYPG17 57799326 Ki = 177 nM T31204 CHB3D6 58405078 Ki = 529 nM T31204 CX2HU7 58405183 Ki = 12 nM T31204 C9UK7P 58438475 IC50 = 4300 nM T31204 C3TGM7 58911532 Ki = 340 nM T31204 CFC79Z 58911534 Ki = 118 nM T31204 CD8JI3 58911579 Ki = 6 nM T31204 CR19FG 58911582 Ki = 139 nM T31204 C4Z5UB 58911604 Ki = 127 nM T31204 C49INW 58911644 Ki = 510 nM T31204 CPC3Z0 58911653 Ki = 40 nM T31204 CNEQ36 58911666 Ki = 1637 nM T31204 CJTR58 58911668 Ki = 930 nM T31204 CG52WR 58911681 Ki = 1340 nM T31204 C2KP7G 59012632 Ki = 14 nM T31204 CRKS62 59312249 EC50 = 1000 nM T31204 CO6P7J 59312265 EC50 > 10000 nM T31204 C31HCO 59312310 EC50 > 10000 nM T31204 C30SVG 60167452 Ki = 1578 nM T31204 CC3Y9Z 67097734 EC50 > 10000 nM T31204 C1LEH8 67268994 Ki = 100 nM T31204 CPV39L 67406727 IC50 = 7600 nM T31204 CKA51D 67781610 Ki = 2.5 nM T31204 C6V0RG 68690817 EC50 > 2500 nM T31204 C1R7EY 68691189 EC50 > 2500 nM T31204 CD3U6K 68731121 Ki > 10000 nM T31204 CZFT98 68803474 EC50 = 794.33 nM T31204 C6IP8Q 69082816 Ki > 10000 nM T31204 CB62XQ 70683433 EC50 = 331 nM T31204 C6FY2A 70687202 Ki = 160 nM T31204 C7QUO3 70687695 EC50 = 304 nM T31204 CZC8S7 70693928 EC50 = 1080 nM T31204 C9P7YD 70695555 Ki = 2600 nM T31204 CVU08A 70695812 Ki = 641 nM T31204 CYAS63 70697549 EC50 = 10 nM T31204 CKD60A 70789640 Ki = 415 nM T31204 C3XNC2 71450247 Ki = 98 nM T31204 C9VZ8J 71450550 Ki = 855 nM T31204 C4TWS5 71452172 Ki = 5097 nM T31204 CTDN12 71452341 Ki = 936 nM T31204 C8YH0J 71455083 Ki = 105 nM T31204 CAQF34 71455625 Ki = 136 nM T31204 CMJ1O9 71457409 Ki > 10000 nM T31204 CS83IF 71459269 Ki = 340 nM T31204 C5DLQ2 71459553 Ki = 204 nM T31204 CK5T4P 71459604 Ki = 2971 nM T31204 C63YLA 71461049 Ki = 29.3 nM T31204 CJD96I 71461050 Ki = 40.4 nM T31204 C5B2WL 71461603 Ki = 15 nM T31204 C4P3JU 71462776 Ki = 162 nM T31204 C3GUQ2 71462777 Ki = 627 nM T31204 CKX5O8 71463061 Ki = 2254 nM T31204 C1DGF4 71499384 IC50 = 7500 nM T31204 C2VP0I 71528204 Ki = 1 nM T31204 CT7UD2 71528205 Ki = 0.97 nM T31204 C8B2VX 71528206 Ki = 0.54 nM T31204 CDL35U 71655748 Ki = 5300 nM T31204 C5LY9W 71681897 Ki = 21 nM T31204 CG34PR 71681898 Ki = 488 nM T31204 CLA5P8 71681899 Ki = 5710 nM T31204 CG4V0A 71682216 Ki = 129 nM T31204 CI46CW 71682217 Ki = 217 nM T31204 C4AMS8 71720492 Ki = 7.1 nM T31204 COWG10 71748255 EC50 > 30000 nM T31204 C3ATN5 72197484 IC50 = 89 nM T31204 CN8A5R 72197486 IC50 = 32 nM T31204 C7AOY4 72198754 IC50 = 43 nM T31204 C4M7KP 72198756 IC50 = 63 nM T31204 CWH6T3 72548703 IC50 = 3.2 nM T31204 C80VRM 72549033 Ki = 144 nM T31204 C78LYM 72698087 Ki = 230 nM T31204 C63HPK 72698088 Ki = 190 nM T31204 CJA8Q5 72713752 IC50 = 64000 nM T31204 C7W4RH 72734860 Ki = 1.8 nM T31204 C8UCZ5 72734861 Ki = 2.1 nM T31204 CZ6SQ7 72734863 Ki = 10 nM T31204 C8JT6B 72734864 Ki = 3.6 nM T31204 CW4IB9 72734866 Ki = 2.4 nM T31204 CY0AE3 72735038 Ki = 1.1 nM T31204 CAZ84Y 72735039 Ki = 86.8 nM T31204 C0MT4E 72735040 Ki = 27.4 nM T31204 C0CK8H 72735041 Ki = 52 nM T31204 CC6Q5R 72771081 Ki < 100 nM T31204 CC65OA 73213195 Ki = 56.23 nM T31204 CW83DK 73213196 Ki = 104 nM T31204 CCV91B 73346042 Ki = 300 nM T31204 CW8A0Y 73349359 Ki = 1965 nM T31204 C6BS5L 73349361 Ki = 2711 nM T31204 C8GQK9 73350823 Ki = 500 nM T31204 CRA5H6 73389570 IC50 = 4000 nM T31204 CPG73S 73417116 EC50 > 5000 nM T31204 C2E7QW 75201901 Ki = 4100 nM T31204 C8IDL3 75306277 Ki = 5.012 nM T31204 CL01RD 76325515 Ki > 10000 nM T31204 C1W5YD 76325516 Ki = 251.19 nM T31204 C0KYJ4 76325517 Ki = 1000 nM T31204 C28RIZ 76518514 Ki = 1381 nM T31204 C4RS7C 83753960 EC50 = 125.89 nM T31204 C70ZVB 86221574 Ki = 79.3 nM T31204 CCY5N2 86302554 Ki > 30000 nM T31204 CP76JG 88912137 Ki = 7568 nM T31204 CWMU25 90644511 IC50 = 67 nM T31204 CG0HF3 91826739 Ki = 1584.89 nM T31204 C0J5YH 91864602 Ki = 232 nM T31204 CCY0O2 100951644 IC50 = 13000 nM T31204 C02GRK 104697662 IC50 = 890 nM T31204 CB0VI8 109052212 IC50 = 90 nM T31204 C5AFD3 112713234 EC50 = 31.62 nM T31204 C8V2SN 116887744 EC50 > 10000 nM T31204 CWR6I1 118112300 IC50 = 3800 nM T31204 CJW1K4 118278424 Ki = 1995.26 nM T31204 C1H3GD 118278480 Ki = 1000 nM T31204 CEMZ15 118464420 Ki = 5.8 nM T31204 C5NSF9 118464421 Ki = 6.3 nM T31204 CV2L6O 118464425 Ki = 38.5 nM T31204 C4C3KD 118464426 IC50 = 35.8 nM T31204 CFNG86 118464427 Ki = 27.5 nM T31204 CON0Q6 118464428 IC50 = 18.1 nM T31204 CQ36GI 118464429 Ki = 1.7 nM T31204 C1CP6Z 118567543 Ki = 754 nM T31204 CSN13R 118706278 Ki = 1.5 nM T31204 CIG56H 118706280 Ki = 1.7 nM T31204 CF5ZR8 118706282 Ki = 0.81 nM T31204 CD1XJ5 118706284 Ki = 0.91 nM T31204 CL4Y6K 118706285 Ki = 1.6 nM T31204 C32KAS 118706287 Ki = 11 nM T31204 C1K5NC 118706290 Ki = 0.67 nM T31204 CGA0O1 118706292 Ki = 6.6 nM T31204 CA0V9U 118706294 Ki = 6.3 nM T31204 C0NSU5 118706296 Ki = 34 nM T31204 CFOE72 118706299 Ki = 0.9 nM T31204 C1DI6Y 118706301 Ki = 4.4 nM T31204 CH3Z8R 118706732 Ki = 1.1 nM T31204 CN4I3G 118706734 Ki = 0.71 nM T31204 CSB25E 118709750 Ki = 270 nM T31204 CD4S9R 118709751 Ki = 520 nM T31204 CUV5Y0 118715454 EC50 > 30000 nM T31204 CI5XK3 118717210 Ki = 41 nM T31204 CYJQ09 118717212 Ki = 31 nM T31204 C1TSR8 118717214 Ki = 3.3 nM T31204 C7YX3Q 118717215 Ki = 4.8 nM T31204 CEZ4M6 118717216 Ki = 2 nM T31204 C1E4GL 118717218 Ki = 0.51 nM T31204 CSJ6N3 118717219 Ki = 1.7 nM T31204 C5LFW4 118717221 Ki = 5.1 nM T31204 CZ65GI 118717222 Ki = 9.1 nM T31204 CU3X0M 118729231 Ki = 40 nM T31204 CNE49D 118729233 Ki = 20 nM T31204 CLD1Z7 118729234 Ki = 170 nM T31204 C4RDW3 118729235 Ki = 650 nM T31204 C47XHR 118729237 Ki = 4100 nM T31204 C08FQG 118729239 Ki = 4100 nM T31204 CR0HA4 118729241 Ki = 540 nM T31204 CY36XK 118729243 Ki = 250 nM T31204 C1VK9B 118729245 Ki = 210 nM T31204 CVR67P 118729247 Ki = 30 nM T31204 CA2Y1F 118729249 Ki = 300 nM T31204 CE1IB3 118729250 Ki = 80 nM T31204 CI8WR2 118729251 Ki = 400 nM T31204 C4ML5K 118729252 Ki = 66 nM T31204 COCH98 118729253 Ki = 70 nM T31204 CQ7K5G 118729255 Ki = 20 nM T31204 C2LDI1 118729257 Ki = 60 nM T31204 COQ04B 118729259 Ki = 200 nM T31204 C9BG0R 118729261 Ki = 8 nM T31204 C63GWU 118729262 Ki = 40 nM T31204 CN24KA 118729263 Ki = 30 nM T31204 C7ZJ2F 118729265 Ki = 50 nM T31204 CL5W0J 118729267 Ki = 70 nM T31204 CN65HD 118729269 Ki = 110 nM T31204 C2B6YA 118729271 Ki = 10 nM T31204 CZ40RY 118729273 Ki = 200 nM T31204 CE38GM 118729275 Ki = 73 nM T31204 CS9W7L 118729277 Ki = 710 nM T31204 C9LI7N 118729278 Ki = 300 nM T31204 C8TEX7 118729279 Ki = 6000 nM T31204 CW3R9X 118729280 Ki = 800 nM T31204 C1D2KW 118733760 EC50 = 2307 nM T31204 CJ1VX4 118733762 EC50 = 86 nM T31204 C2YQC3 118733764 EC50 = 3004 nM T31204 CSE5K7 118733766 EC50 = 3436 nM T31204 C8FZI7 118733776 EC50 = 3034 nM T31204 C4U6XR 118733778 EC50 = 5012 nM T31204 C4V6FB 118733780 EC50 = 5300 nM T31204 CSZ6Q7 118733792 EC50 = 4411 nM T31204 CQZ71R 118733794 EC50 = 4602 nM T31204 CC6H7T 118733796 EC50 = 6877 nM T31204 C7MRW8 118733798 EC50 = 1688 nM T31204 CT4BW7 118733800 EC50 = 6094 nM T31204 C7ZS0V 118733802 EC50 = 422 nM T31204 CWM78D 118733804 EC50 = 4521 nM T31204 C6VO5G 118733806 EC50 = 632 nM T31204 C7RUF2 118733808 EC50 = 1485 nM T31204 CNH6K2 118733810 EC50 = 839 nM T31204 C0SH9U 118733812 EC50 = 6166 nM T31204 CXAZ36 118733814 EC50 = 4911 nM T31204 C1CXD4 118733816 EC50 = 735 nM T31204 CSN70M 118733818 EC50 = 1994 nM T31204 CX3H6M 118736623 EC50 = 1484 nM T31204 C61ABM 118736624 EC50 = 18 nM T31204 CR4ZF9 118736626 EC50 = 22 nM T31204 C8TE3L 118736627 EC50 = 27 nM T31204 C3XJY0 118736628 EC50 = 33 nM T31204 C7BMI8 118736630 EC50 = 30 nM T31204 CP54MG 118736631 EC50 = 27 nM T31204 CX31UR 122182283 Ki = 1258.93 nM T31204 CRJE23 122185011 IC50 = 250 nM T31204 C5X8MN 122186880 Ki = 96 nM T31204 CKZ3J7 122186881 Ki = 209 nM T31204 CJ26IS 122187375 Ki = 307 nM T31204 CJG0W7 122187376 Ki = 601 nM T31204 C0K9WV 122187377 Ki = 663 nM T31204 C7RP0M 122187378 Ki = 299 nM T31204 CY42PC 122187379 Ki = 416 nM T31204 C90PRI 122187381 Ki = 715 nM T31204 C1Z7CU 122187382 Ki = 419 nM T31204 CQE18J 122187383 Ki = 1429 nM T31204 CHVR64 122188579 Ki = 2500 nM T31204 C7ODW3 122195524 Ki > 900 nM T31204 C8K9XA 122196341 IC50 = 220 nM T31204 CLW53P 122483274 Ki = 83 nM T31204 CO63ET 122483280 Ki = 93 nM T31204 C4QM2E 124247485 Ki = 97 nM T31204 CCM0S8 126844990 EC50 = 2344.23 nM T31204 CTBN56 127026052 Ki = 16.6 nM T31204 CBE56W 127026514 Ki = 419 nM T31204 C0SZI4 127026515 Ki = 101 nM T31204 CAX87V 127026556 EC50 = 2182 nM T31204 C4PW9X 127026867 EC50 = 927 nM T31204 CW40RC 127028088 EC50 = 208.93 nM T31204 C7X4RJ 127028094 EC50 = 1000 nM T31204 C7A8OC 127028095 EC50 = 165 nM T31204 CGA51D 127028100 EC50 = 30.9 nM T31204 C90QPM 127028101 EC50 = 101 nM T31204 C0SGM2 127028405 EC50 = 25 nM T31204 CE0T8G 127028406 EC50 = 27 nM T31204 C3H9NU 127028407 EC50 = 453 nM T31204 C8MC1I 127028408 Ki = 68 nM T31204 C9YU1E 127028422 EC50 = 714 nM T31204 CPF1T5 127028423 EC50 = 30 nM T31204 CA9IP6 127028732 EC50 = 954.99 nM T31204 CG7OW2 127029036 EC50 = 3311.31 nM T31204 CC4U8R 127029581 EC50 = 501.19 nM T31204 C6O2SL 127034715 Ki = 4.1 nM T31204 CNO80F 127034729 Ki = 59 nM T31204 CB02LG 127034730 Ki = 231 nM T31204 CZ61LK 127034966 IC50 > 5011.87 nM T31204 CA0SN5 127034967 EC50 > 5011.87 nM T31204 CQ0ZT9 127035062 Ki = 26 nM T31204 CW1KD7 127035063 Ki = 5.8 nM T31204 CO3W6A 127035064 Ki = 4.6 nM T31204 CTY04X 127035065 Ki = 6.8 nM T31204 CPM2B8 127035066 Ki = 36 nM T31204 CU49VE 127036186 Ki = 60.26 nM T31204 CP04WI 127036910 Ki = 59 nM T31204 CG06BD 127036932 Ki = 30.2 nM T31204 CVW71O 127036953 Ki = 52.48 nM T31204 C0HLY8 127037059 Ki = 21 nM T31204 CZ6QR4 127037093 Ki = 17 nM T31204 CS9V0E 127048333 Ki = 1.7 nM T31204 CQM81O 127048334 Ki = 3.1 nM T31204 CJG5E2 127048335 Ki = 3.4 nM T31204 CUK40V 127048336 Ki = 13 nM T31204 CC7BU0 127049059 Ki = 905 nM T31204 C42FHY 127049060 Ki = 202 nM T31204 C6SP9O 127049979 Ki = 54 nM T31204 C1CB0Z 127049980 Ki = 45 nM T31204 C0JUA9 127049981 Ki = 51 nM T31204 C69RCG 127049982 Ki = 18 nM T31204 C0M9PE 127049983 Ki = 17 nM T31204 CI5XG2 127050282 Ki = 14 nM T31204 CX53AC 127050632 Ki = 36 nM T31204 CX5H1W 127051482 Ki = 14 nM T31204 CTL0S1 127051516 Ki = 122 nM T31204 CTL8J1 127051843 Ki = 151.36 nM T31204 CF6V9Q 127051844 Ki = 587 nM T31204 C8TNB1 127051845 Ki = 723 nM T31204 C5ONG1 127051864 Ki = 338.84 nM T31204 CVQW26 127051865 Ki = 758 nM T31204 CRF85X 127052458 Ki = 354.81 nM T31204 CCY71I 127052465 Ki = 398.11 nM T31204 CPO4C3 127052468 Ki = 1247 nM T31204 CSQ2N8 127052486 Ki = 512.86 nM T31204 C4YJ8H 127052487 Ki = 51 nM T31204 CLU7C1 127052757 Ki = 1698.24 nM T31204 C95KYT 127052758 Ki = 561 nM T31204 CYNR02 127052759 Ki = 204 nM T31204 C6XR8U 127053028 Ki = 18 nM T31204 C7MQK8 127053042 Ki = 1166 nM T31204 C50GOC 130442480 Ki = 6700 nM T31204 CM04RF 130442572 Ki = 830 nM T31204 C5XZN0 132007291 Ki = 4000 nM T31204 C1RI8Q 132060720 Ki = 389.5 nM T31204 CY8B9L 132060743 Ki = 1117 nM T31204 CGHO19 132060770 Ki = 505 nM T31204 CT81OY 132060776 Ki = 894 nM T31204 CFXL21 132060812 Ki = 65 nM T31204 C7CSU4 132075278 Ki = 360 nM T31204 CDB85P 132559161 Ki = 770 nM T31204 CAVB41 132584404 Ki > 10000 nM T31204 CP26SI 132820207 EC50 = 630.96 nM T31204 CYBK37 132820208 EC50 = 398.11 nM T31204 CEY94B 132820209 EC50 = 1258.93 nM T31204 CC7PW1 132820210 EC50 = 630.96 nM T31204 CN08ZY 132820211 EC50 = 100 nM T31204 C78MPD 132820212 EC50 = 158.49 nM T31204 C8O2EP 134130246 Ki = 18 nM T31204 CM10CR 134132665 EC50 = 794.33 nM T31204 CQX4U3 134133064 Ki = 524.81 nM T31204 CGH25V 134133531 EC50 = 2511.89 nM T31204 C0J2ML 134133604 Ki = 109 nM T31204 CM0TS6 134133967 Ki = 239 nM T31204 CYRW09 134133994 EC50 > 10000 nM T31204 CP3J9C 134134314 Ki = 6.31 nM T31204 CZ8HL0 134134668 Ki = 476 nM T31204 C6G4CW 134135745 Ki = 163 nM T31204 CGX03A 134136246 Ki = 147.91 nM T31204 CZ0RN8 134136722 EC50 > 1000 nM T31204 CBOH57 134136932 EC50 = 1000 nM T31204 CS1HT4 134137343 EC50 = 63.1 nM T31204 CE93ZP 134137441 EC50 = 199.53 nM T31204 CEU49D 134137640 EC50 > 1000 nM T31204 C9A6KG 134138183 Ki = 186 nM T31204 C5JP1R 134138627 EC50 = 7.943 nM T31204 CH0FX4 134138769 Ki = 77 nM T31204 C0XHJ2 134139670 EC50 = 501.19 nM T31204 CR7C9U 134139964 Ki = 39.81 nM T31204 CNSB82 134141050 Ki = 1480 nM T31204 C86RBW 134141127 EC50 = 1.995 nM T31204 CLW86T 134141354 Ki = 501 nM T31204 C4ECW0 134141640 EC50 = 630.96 nM T31204 C68AXD 134141831 Ki = 11.1 nM T31204 CCS9A1 134142903 Ki = 63.1 nM T31204 CJFV62 134143302 Ki = 332 nM T31204 C08RJA 134143536 Ki = 34 nM T31204 C5L9BD 134143752 Ki = 1.8 nM T31204 CV8IR0 134143977 Ki = 12.59 nM T31204 C1NDF5 134144277 EC50 = 6309.57 nM T31204 CR5L4K 134144303 Ki = 549 nM T31204 C71PIY 134144970 Ki = 45 nM T31204 CC9P2T 134146194 Ki = 64 nM T31204 C19LRO 134146585 Ki = 2100 nM T31204 CUQ0F6 134147456 Ki = 25.12 nM T31204 CZPS45 134148291 EC50 = 630.96 nM T31204 C7S5RQ 134149008 Ki = 4700 nM T31204 CBU81N 134149168 Ki = 1905 nM T31204 COUJ52 134149355 Ki = 125.89 nM T31204 CAO9T6 134150123 Ki = 671 nM T31204 CM31CH 134150311 EC50 > 1000 nM T31204 CLU34D 134151427 Ki = 391 nM T31204 CFV6S8 134151626 EC50 = 1258.93 nM T31204 C8PT9W 134152052 Ki = 4.4 nM T31204 C73ISY 134152157 Ki = 73 nM T31204 CL0G3W 134152924 EC50 = 79.43 nM T31204 CT16QG 134153263 EC50 > 10000 nM T31204 CB6M5Y 134153538 Ki = 323.59 nM T31204 CP41RT 134154065 Ki = 3.2 nM T31204 C79TEI 134154068 Ki = 15.49 nM T31204 CMJ1U3 134154387 Ki = 125.89 nM T31204 C4VGJ5 134154679 Ki = 7 nM T31204 C6QAY2 134155116 Ki = 294 nM T31204 CZFB29 134155462 Ki = 4800 nM T31204 CE64VO 134155579 EC50 = 100 nM T31204 CZJ15H 134155852 Ki = 25.12 nM T31204 C87HWQ 134155992 EC50 = 7943.28 nM T31204 CVR87Q 134156222 Ki = 478.63 nM T31204 C7UOJ8 134156506 Ki = 163 nM T31204 C1IF0S 134156657 EC50 = 39.81 nM T31204 C5UQW2 134157367 Ki = 534 nM T31204 CF7EV5 134265590 EC50 = 779 nM T31204 CL5FW8 134265616 EC50 = 165 nM T31204 CR06XB 134265618 EC50 = 4020 nM T31204 CNA08H 134265620 EC50 = 758 nM T31204 C46YNU 134265622 EC50 = 478 nM T31204 CA5PX2 134265627 EC50 = 115 nM T31204 CAS9Z4 134265663 EC50 = 21.7 nM T31204 CW3I6K 134265665 EC50 = 1290 nM T31204 CVY5G8 134265675 EC50 = 307 nM T31204 C6SLE4 134265705 EC50 = 61.2 nM T31204 C8WAR6 134265732 EC50 = 1290 nM T31204 C1GY2T 135156251 EC50 > 10000 nM T31204 C6N8GM 135367405 Ki = 106 nM T31204 C6LU0C 135367816 Ki = 247 nM T31204 CD2TH9 135367820 Ki = 505 nM T31204 C5AMD9 135367857 Ki = 150 nM T31204 C8WL0I 135449090 Ki = 4554 nM T31204 CTE23K 135464118 Ki = 51 nM T31204 CB53EI 135465870 Ki = 716 nM T31204 C7AGR0 135474338 Ki = 190 nM T31204 C34FXW 135501716 Ki = 1676 nM T31204 C1CZ9M 135514796 Ki = 232 nM T31204 C03HVY 135846955 Ki = 1284 nM T31204 CQCT18 135846958 Ki = 1378 nM T31204 CE4QG5 135846981 Ki = 5055 nM T31204 C3UB7L 135846982 Ki = 1274 nM T31204 CUKO20 136020617 Ki = 505 nM T31204 COF0U5 136020618 Ki = 130 nM T31204 CBV06G 136020620 Ki = 1541 nM T31204 CF89JI 136030596 Ki = 1360 nM T31204 CE8GB9 136030693 Ki = 1260 nM T31204 C65VFI 136030744 Ki = 3922 nM T31204 COIX80 136054961 Ki = 1000 nM T31204 CA3JC8 136118613 Ki = 228 nM T31204 CQ2GP6 136118614 Ki = 94 nM T31204 C6R4IC 136118615 Ki = 593 nM T31204 CS0JL5 136118616 Ki = 99 nM T31204 C8RH6M 136118617 Ki = 883 nM T31204 CN4U6K 136118618 Ki = 489 nM T31204 CHWC38 136118619 Ki = 661 nM T31204 C5UDW3 136118620 Ki = 589 nM T31204 C8I6UN 136118621 Ki = 349 nM T31204 CV4E6W 136118635 Ki = 369 nM T31204 CFI2X7 136118636 Ki = 2714 nM T31204 C0UH1B 136118638 Ki = 780 nM T31204 C6G4AY 136118639 Ki = 1346 nM T31204 C40VES 136118640 Ki = 1136 nM T31204 CH4Q8O 136118646 Ki = 993 nM T31204 C43JTG 136118647 Ki = 287 nM T31204 CLH0V9 136118648 Ki = 50 nM T31204 C76XEJ 136118649 Ki = 93 nM T31204 CN0V5C 136118650 Ki = 154 nM T31204 CR72MQ 136118651 Ki = 353 nM T31204 CD7OE2 136118652 Ki = 774 nM T31204 CG5TX8 136118653 Ki = 520 nM T31204 CCHM67 136118657 Ki = 839 nM T31204 C0W1TM 136118658 Ki = 897 nM T31204 C40LYH 136118659 Ki = 1620 nM T31204 CZ7C3Y 136118660 Ki = 2468 nM T31204 C42FCS 136118661 Ki = 965 nM T31204 CR3DK1 136118716 Ki = 447 nM T31204 CON04G 136118728 Ki = 269 nM T31204 COX1F8 136118729 Ki = 457 nM T31204 CY5GU4 136118730 Ki = 784 nM T31204 C0R5PV 136118732 Ki = 1422 nM T31204 CAE39V 136188797 Ki = 3900 nM T31204 CLAP52 136259032 Ki = 1500 nM T31204 C8SI2Q 136928971 IC50 = 49.4 nM T31204 CGS61F 137553161 Ki = 153 nM T31204 CBX2V5 137631812 EC50 > 10000 nM T31204 CQO58W 137632042 EC50 > 10000 nM T31204 CDQ6X3 137632069 EC50 > 10000 nM T31204 C64KPN 137632218 EC50 > 10000 nM T31204 CMO30D 137633009 EC50 > 10000 nM T31204 C5ZL0C 137633983 EC50 > 10000 nM T31204 CATU84 137634233 EC50 > 10000 nM T31204 CXCJ60 137634432 EC50 > 10000 nM T31204 C9M3RV 137635151 EC50 = 87 nM T31204 C94MFJ 137635172 EC50 > 10000 nM T31204 C5N4PR 137635711 EC50 > 10000 nM T31204 CJT0A2 137635932 EC50 > 10000 nM T31204 CPQ34V 137636430 EC50 > 10000 nM T31204 CQ71WO 137636435 EC50 > 10000 nM T31204 C8Z1XW 137636480 EC50 = 112.2 nM T31204 C4OT7C 137637069 EC50 > 5000 nM T31204 CTD64R 137637165 EC50 > 10000 nM T31204 CK29VL 137637650 EC50 > 10000 nM T31204 C71BUE 137637880 EC50 = 238 nM T31204 C56GTL 137638508 EC50 > 10000 nM T31204 CM0DJ5 137638903 EC50 > 10000 nM T31204 CK8UC2 137639485 EC50 > 10000 nM T31204 CEQ68W 137639630 EC50 > 10000 nM T31204 CPQ83I 137639705 EC50 > 10000 nM T31204 C5KX6V 137640062 Ki = 411 nM T31204 C62QAM 137640945 EC50 = 807 nM T31204 C90GKM 137641125 EC50 > 5000 nM T31204 CUQ8F5 137641376 EC50 > 10000 nM T31204 C6P9FW 137642149 EC50 > 10000 nM T31204 CO6J9Q 137642857 EC50 > 10000 nM T31204 CPL0K5 137643658 EC50 > 10000 nM T31204 C1ZP9R 137643846 EC50 = 56 nM T31204 CIKD85 137644487 EC50 > 10000 nM T31204 CRGN16 137644935 EC50 = 641 nM T31204 CSO38A 137645024 EC50 > 5000 nM T31204 CPCY48 137645406 Ki = 2144 nM T31204 CRU20V 137645667 EC50 > 10000 nM T31204 CA7P4F 137645674 EC50 > 10000 nM T31204 CUR7T5 137645858 EC50 > 10000 nM T31204 C5Q6DL 137646111 EC50 > 10000 nM T31204 CPI68E 137646281 Ki = 42 nM T31204 C9EYB1 137646716 EC50 > 10000 nM T31204 C2O1XW 137646874 EC50 > 10000 nM T31204 C6C3IK 137646921 EC50 > 10000 nM T31204 CN5R7Q 137647004 EC50 > 10000 nM T31204 CD2TE0 137647007 EC50 > 10000 nM T31204 C5Y0FG 137647246 EC50 > 10000 nM T31204 CU6V5W 137647439 EC50 = 89 nM T31204 CA48GB 137647635 EC50 = 48 nM T31204 CQA0B2 137647926 EC50 > 10000 nM T31204 C4HX6J 137648810 EC50 > 10000 nM T31204 C1GZV3 137650863 EC50 = 95.5 nM T31204 CXV3D7 137651249 EC50 > 10000 nM T31204 C1SY4J 137651715 EC50 > 5000 nM T31204 CTE69H 137652480 EC50 > 10000 nM T31204 CY59NZ 137652713 EC50 > 10000 nM T31204 CC12VB 137653689 EC50 > 10000 nM T31204 CKT1F5 137654351 EC50 > 10000 nM T31204 CS1Y8F 137654798 EC50 > 10000 nM T31204 CZ50SL 137654926 EC50 > 10000 nM T31204 CJMR75 137655187 EC50 = 331.13 nM T31204 C53QIZ 137655324 EC50 = 24 nM T31204 CHI8M2 137655535 EC50 > 10000 nM T31204 CB20MW 137655657 EC50 = 274 nM T31204 C91UBP 137655705 EC50 > 10000 nM T31204 C1PKE6 137655741 EC50 > 10000 nM T31204 CKW87Y 137655846 EC50 > 10000 nM T31204 C60XIF 137655882 EC50 > 10000 nM T31204 C17NVY 137656030 EC50 > 10000 nM T31204 CL8RT7 137656524 EC50 > 10000 nM T31204 CKQ7Y9 137658074 EC50 > 10000 nM T31204 C0OI2B 137658246 EC50 > 10000 nM T31204 CH9R5V 137658409 EC50 > 5000 nM T31204 C3JG5Z 137659281 EC50 > 10000 nM T31204 CAM68B 137660072 EC50 > 10000 nM T31204 C5Q9CM 137660307 EC50 = 570 nM T31204 C3UHP5 137660422 EC50 > 10000 nM T31204 C6SHF4 137661018 EC50 > 10000 nM T31204 C0YZF2 137661221 EC50 > 10000 nM T31204 C8JH6R 137661673 EC50 = 3 nM T31204 CN52AG 137662193 EC50 > 10000 nM T31204 CAP26G 139030523 Ki = 219 nM T31204 C7KC3T 145963830 Ki = 100 nM T31204 CHDN35 145964150 Ki = 7500 nM T31204 C1KH2E 145964159 Ki = 47 nM T31204 C12OVL 145965034 Ki > 10000 nM T31204 CKO51D 145965628 Ki = 1100 nM T31204 C5W4LM 145965940 Ki = 810 nM T31204 C4EQ9C 145966293 EC50 = 489 nM T31204 C81VUO 145967771 Ki = 620 nM T31204 CJS56K 145967795 Ki = 1500 nM T31204 CQJ5O8 145971635 Ki > 10000 nM T31204 C7BVC1 145972374 Ki = 1000 nM T31204 C79TNE 145972796 Ki = 1200 nM T31204 CT5CX0 145973771 Ki = 2780 nM T31204 C6XIN0 145974114 Ki > 10000 nM T31204 CD8ZL6 145974750 Ki = 400 nM T31204 C6PH4F 145975226 Ki = 1400 nM T31204 C71CYU 145975946 Ki = 4300 nM T31204 C2TN8W 145976085 Ki = 380 nM T31204 C7L9DG 145976983 Ki = 1400 nM T31204 C6BFY7 145977338 Ki = 100 nM T31204 C0Y6QO 145977799 Ki = 690 nM T31204 C3BI1R 145978113 Ki = 3000 nM T31204 CQU8R0 145978665 Ki = 2400 nM T31204 C6AV9G 145978819 Ki = 1400 nM T31204 CI8SJ4 145979048 IC50 = 1962.5 nM T31204 C87MSW 145980271 Ki = 509 nM T31204 C58OUC 145981805 Ki = 3 nM T31204 CNJH37 145986752 Ki = 729 nM T31204 C86XQR 145988313 Ki = 4.5 nM T31204 CUGO10 145988693 Ki = 177 nM T31204 CN69QU 145989393 IC50 = 74.9 nM T31204 C03BKU 145989551 Ki = 16.6 nM T31204 C4GV8Q 145990586 Ki = 246 nM T31204 C30NLA 145990659 Ki = 313.5 nM T31204 CCP2U1 145992489 Ki = 2199 nM T31204 CQ93KE 145993540 Ki = 3.36 nM T31204 CCUJ49 145993660 IC50 = 215 nM T31204 CC2G1V 146025727 Ki = 1100 nM T31204 CG97ER 146709966 Ki = 2.512 nM T31204 C6FX4M 147636204 Ki > 10000 nM T31204 CW4S2X 147652368 Ki > 10000 nM T31204 CF5B2L 147653864 Ki = 19.95 nM T31204 C5PNX8 148302367 Ki = 125.89 nM T31204 C2E5HK 149396365 Ki = 125.89 nM T31204 C9T0PS 153061504 Ki = 19.95 nM T31204 CF7J3M 153287535 Ki = 1000 nM T31204 C72MVW 153287537 Ki > 10000 nM T31204 CAF36V 153287539 Ki = 251.19 nM T31204 C1FA0K 153287541 Ki = 251.19 nM T31204 CEQ69Z 153287542 Ki = 158.49 nM T31204 C9A7SV 153287550 Ki > 10000 nM T31204 C91KST 153287551 Ki = 501.19 nM T31204 C6P3SR 153287553 Ki = 501.19 nM T31204 C3G5CJ 153287557 Ki = 316.23 nM T31204 CW31CT 153287566 Ki = 199.53 nM T31204 CYP86E 153287567 Ki = 316.23 nM T31204 CS73ZC 153287568 Ki = 79.43 nM T31204 CV9G7Z 153287572 Ki = 177.83 nM T31204 CO85KL 153287574 Ki = 794.33 nM T31204 CU4H6L 155512064 Ki = 2681 nM T31204 CCD9N1 155512086 Ki = 214 nM T31204 CUSA24 155519891 Ki = 251.19 nM T31204 CGS21U 155525549 Ki > 10000 nM T31204 CP76JX 155526977 Ki = 251.19 nM T31204 CRF1A0 155527638 EC50 = 1.259 nM T31204 C8QF4Y 155529999 EC50 = 800 nM T31204 CS2BT0 155530292 Ki = 1570 nM T31204 CFC74M 155531067 Ki = 212 nM T31204 CV6ST2 155531084 Ki = 422 nM T31204 CX43DV 155532107 EC50 = 2 nM T31204 C6KAU3 155534798 Ki = 2900 nM T31204 COT9U8 155535203 Ki = 2900 nM T31204 C05NHQ 155535754 Ki = 742 nM T31204 C7OIP3 155535969 EC50 = 903 nM T31204 CB79ZW 155536080 Ki = 144.54 nM T31204 CIUS98 155536619 Ki = 1910 nM T31204 C9S2IA 155539605 Ki = 231 nM T31204 C4FJL0 155539960 EC50 = 114.82 nM T31204 C72KHI 155540514 EC50 = 21.88 nM T31204 C1JM5R 155540523 Ki = 552 nM T31204 CMT60C 155543832 Ki = 1520 nM T31204 CGU5M0 155544723 Ki = 3044 nM T31204 CSX3M0 155548666 EC50 = 562.34 nM T31204 C9BAV3 155549312 EC50 = 450 nM T31204 C7KWB9 155550387 Ki = 102 nM T31204 CN39VC 155551164 EC50 = 281.84 nM T31204 CHYA95 155554410 Ki = 2051 nM T31204 C0PBT3 155555147 Ki > 10000 nM T31204 C3DF2T 155556596 Ki = 51 nM T31204 CBS89O 155556618 Ki = 2010 nM T31204 CJBX01 155557042 Ki = 630.96 nM T31204 C4XRZ1 155558626 Ki = 209 nM T31204 C4AG0H 155558726 Ki = 8200 nM T31204 C2Q6KU 155558968 Ki = 840 nM T31204 C5L8HB 155560629 EC50 = 11.75 nM T31204 C9LV7U 155561048 EC50 = 363 nM T31204 CH0VC3 155561439 Ki = 1210 nM T31204 CSK27Q 155561712 Ki = 106 nM T31204 C9P7AU 155562772 EC50 = 410 nM T31204 C4N9GU 155563428 Ki = 97 nM T31204 CR12DI 155565189 Ki = 870 nM T31204 CFNC10 155565326 Ki = 718 nM T31204 CBI7N3 155566272 Ki = 334 nM T31204 C6DQ1K 155566338 Ki = 472 nM T31204 CPW8M5 155567457 Ki = 1860 nM T31204 C3N9VU 10251906 Ki = 231 nM T31204 CQ1LV7 135508617 Ki = 1248 nM T31204 CGK7B1 135511529 Ki = 964 nM T31204 CRKP76 136016509 Ki = 852 nM T31204 D00APD 15124 Ki = 6300 nM T31204 D00AVR 135476741 Ki = 4449 nM T31204 D00EMF 3644637 Ki = 100 nM T31204 D00GOY 6604042 EC50 = 11 nM T31204 D00YVE 10219723 EC50 = 40 nM T31204 D01BGW 11708275 Ki = 7.5 nM T31204 D01KAX 135453290 Ki = 8.1 nM T31204 D01NOZ 16665072 IC50 = 1500 nM T31204 D01NTM 11264955 EC50 = 4.1 nM T31204 D01SJL 135509961 Ki = 3.8 nM T31204 D01TSX 9840090 Ki = 18 nM T31204 D01WWC 16573 Ki = 323 nM T31204 D01XZI 10015055 Ki = 240 nM T31204 D02YNH 9901086 EC50 = 65.3 nM T31204 D03DET 10287730 Ki = 1258.93 nM T31204 D03DLZ 6089 Ki = 101 nM T31204 D03WTU 5886965 IC50 = 2600 nM T31204 D04TPO 16006492 IC50 > 400 nM T31204 D04YCJ 135399866 Ki = 1.7 nM T31204 D05EQG 5265 Ki = 1258.93 nM T31204 D05NWH 443390 Ki = 10 nM T31204 D05SWY 44404899 Ki = 1242 nM T31204 D05XGR 6918647 Ki = 630.96 nM T31204 D05ZUX 44207909 Ki >= 1000 nM T31204 D06ABJ 11492162 Ki = 8.39 nM T31204 D06VDN 443391 Ki = 100 nM T31204 D07LRJ 5312149 Ki < 3981.07 nM T31204 D07RIQ 71028 Ki = 491 nM T31204 D07XTU 1229 Ki = 1.6 nM T31204 D08CKM 9863250 Ki < 2511.89 nM T31204 D08EFH 36906 Ki = 7.8 nM T31204 D08GJS 44404906 Ki = 745 nM T31204 D08ZWM 4980 EC50 = 58 nM T31204 D09BNS 439280 EC50 = 1 nM T31204 D09HJL 10331436 Ki = 5.3 nM T31204 D09OYA 2107 Ki = 13 nM T31204 D09RPR 16737207 Ki > 10000 nM T31204 D09WIL 10028436 Ki = 91.2 nM T31204 D0A0GU 44247568 Ki = 328 nM T31204 D0AP6N 44404886 Ki = 5.8 nM T31204 D0C5XQ 1832 Ki = 52 nM T31204 D0DY5G 443389 Ki = 12.59 nM T31204 D0E3AL 56597938 Ki = 0.6 nM T31204 D0E6NW 9859257 EC50 = 3 nM T31204 D0F5WP 135520431 Ki = 15 nM T31204 D0F6CD 5202 EC50 = 0.5 nM T31204 D0G8CV 9954003 Ki = 1 nM T31204 D0H3WJ 44435193 Ki = 170 nM T31204 D0H5XR 3045225 Ki = 2.5 nM T31204 D0H7PC 6918553 Ki > 3981.07 nM T31204 D0H9QG 5312148 Ki < 5011.87 nM T31204 D0I9RW 135427931 Ki = 6 nM T31204 D0J2UA 135433933 Ki = 2671 nM T31204 D0J3PJ 4331799 Ki = 320 nM T31204 D0J6JT 1355 Ki = 10 nM T31204 D0K5NZ 68848 Ki = 1.995 nM T31204 D0KH5R 10449757 IC50 = 13 nM T31204 D0KS0I 24894910 EC50 > 10000 nM T31204 D0L5MW 181743 Ki = 543 nM T31204 D0L8MR 4076 Ki = 795.1 nM T31204 D0M1YU 10198431 EC50 = 1.1 nM T31204 D0N6OL 11452268 IC50 = 1900 nM T31204 D0N8YG 135414348 Ki = 8.7 nM T31204 D0O5KK 44451373 Ki = 34 nM T31204 D0O7MW 14702424 Ki = 1617 nM T31204 D0PC7A 10106214 Ki = 94 nM T31204 D0R3GW 10296414 Ki = 1584.89 nM T31204 D0R8VT 44404883 Ki = 38 nM T31204 D0T2RY 9948320 Ki >= 1000 nM T31204 D0T7RY 9813197 Ki = 100 nM T31204 D0T8UR 44404904 Ki = 1242 nM T31204 D0U7BH 9815618 EC50 = 15.85 nM T31204 D0U9HE 3693566 Ki = 316.23 nM T31204 D0UZ4J 6604926 Ki = 3981.07 nM T31204 D0W8EB 44404905 Ki = 98 nM T31204 D0XX7J 44451369 Ki = 90 nM T31204 D0Y0SA 135399666 Ki = 35 nM T31204 D0Z7GS 43922 Ki = 2495 nM T31204 D0ZZ4Z 21854226 Ki = 423 nM T62548 D06GDY 43815 IC50 = 1100 nM T62548 D0E3TC 44259 IC50 = 1440 nM T62548 D00YYO 118888942 IC50 = 220 nM T62548 D05PTF 118888905 IC50 = 2700 nM T62548 D0U5IW 118888913 IC50 = 25000 nM T62548 D0WX0K 71680628 IC50 = 530 nM T62548 D0YD7S 118888923 IC50 = 4800 nM T62548 D0R2TM 5287736 IC50 = 42 nM T62548 CW02OU 14978 Ki = 67000 nM T62548 C75EDQ 644355 IC50 > 100000 nM T62548 C5HPF3 644356 IC50 > 100000 nM T62548 CLJ97Z 963518 IC50 = 5700 nM T62548 C86HDP 1959269 IC50 > 10000 nM T62548 CT7L1J 2766553 IC50 = 4400 nM T62548 CHF4O5 4356253 IC50 = 1200 nM T62548 C5KBV9 5078538 IC50 = 563000 nM T62548 C9NBG7 5330546 IC50 > 100000 nM T62548 C95WKV 5353430 IC50 = 126000 nM T62548 CI26XO 6910830 IC50 > 10000 nM T62548 C4TJ9V 9579814 IC50 = 1800 nM T62548 CA80PO 9661728 IC50 = 700 nM T62548 CO08EA 9714186 IC50 > 10000 nM T62548 CEB53H 9724880 IC50 = 49 nM T62548 C48HIZ 11155477 IC50 = 1.2 nM T62548 CM6DO0 11233873 IC50 = 770 nM T62548 CQR05P 11494718 EC50 = 41000 nM T62548 CHT93E 11502159 IC50 = 9.9 nM T62548 CNQ61U 11524891 IC50 = 6.8 nM T62548 CUW0C5 11567501 IC50 = 19 nM T62548 CWRY72 11567821 IC50 = 12 nM T62548 C4WCL9 11603404 IC50 = 24 nM T62548 C6LDN4 11617898 IC50 = 14 nM T62548 C7WZY3 16066456 IC50 = 41 nM T62548 C7YG1N 24759534 IC50 = 610 nM T62548 CB3Z8Q 25210972 IC50 = 20000 nM T62548 C16ISR 25218571 IC50 = 6300 nM T62548 CP81DI 25218601 IC50 = 7900 nM T62548 C6ND4K 43839983 IC50 = 100 nM T62548 CG4DJ2 43839997 IC50 = 440 nM T62548 CG89VQ 44256165 IC50 = 3190 nM T62548 CF8U5T 44256167 IC50 = 6320 nM T62548 C0SE3Q 44256203 IC50 = 5520 nM T62548 CT2MO1 44256205 IC50 = 8270 nM T62548 CI21MW 44256238 IC50 = 1650 nM T62548 CUM54B 44256240 IC50 = 6430 nM T62548 CZ7V6J 44256242 IC50 = 4900 nM T62548 CX9NJ8 44256244 IC50 = 13000 nM T62548 CWK6F0 44256275 IC50 = 3060 nM T62548 CU03ZE 44256279 IC50 = 10100 nM T62548 CE3Y6K 44256281 IC50 = 5300 nM T62548 C1QXF2 44256314 IC50 = 9300 nM T62548 C2MS6Q 44256343 IC50 = 11500 nM T62548 C2IJ6R 44256345 IC50 = 2260 nM T62548 CN35VU 44256347 IC50 = 5700 nM T62548 C7NB5X 44256371 IC50 = 4220 nM T62548 CV1X8T 44256373 IC50 = 6200 nM T62548 C6UKT1 44256406 IC50 > 10000 nM T62548 CO89LE 44256480 IC50 > 10000 nM T62548 CUT0N9 44308442 IC50 = 557000 nM T62548 C60ZSA 58897672 IC50 = 5600 nM T62548 CXJ63M 59603829 IC50 = 23000 nM T62548 CQEU96 59603842 IC50 = 160 nM T62548 C61EBT 60141028 IC50 > 10000 nM T62548 CFQ1U4 60142431 IC50 = 3060 nM T62548 C18CIG 60142559 IC50 = 1720 nM T62548 C6DHB7 60142693 IC50 = 2630 nM T62548 C1FOD2 60142694 IC50 = 8300 nM T62548 CAXK87 60142952 IC50 > 10000 nM T62548 CBCE37 60142954 IC50 = 2140 nM T62548 CL0N9F 60143086 IC50 = 13000 nM T62548 CZT65A 60143089 IC50 = 9700 nM T62548 CV63UL 67240318 IC50 > 10000 nM T62548 C5DGR9 69036886 IC50 = 10000 nM T62548 CN8F4V 70690082 IC50 > 10000 nM T62548 CPZ67U 71315739 IC50 = 63100 nM T62548 CR5N7S 72724699 IC50 > 10000 nM T62548 C3R6FU 72724978 IC50 > 10000 nM T62548 C25OTJ 72725039 IC50 > 10000 nM T62548 C3I4GZ 72725092 IC50 = 4050 nM T62548 CFEA16 72725094 IC50 = 11900 nM T62548 CRWU68 72725096 IC50 > 10000 nM T62548 CS7I6A 72725098 IC50 = 17000 nM T62548 C8XK0I 72725161 IC50 > 10000 nM T62548 C3LF8A 72725163 IC50 = 8100 nM T62548 CA6WD3 72725165 IC50 = 3800 nM T62548 C3KWN2 72725221 IC50 = 660 nM T62548 C6L5TE 72725225 IC50 = 3190 nM T62548 C6UFA2 72725284 IC50 = 6050 nM T62548 CN8X5K 72725286 IC50 = 3200 nM T62548 CQH30J 72725289 IC50 = 960 nM T62548 CWUN78 72725404 IC50 = 3970 nM T62548 C78TKB 72725451 IC50 > 10000 nM T62548 C1NI9K 72725453 IC50 > 10000 nM T62548 CSY5U6 72725501 IC50 = 9160 nM T62548 CGNJ85 72725616 IC50 = 850 nM T62548 C7T6EA 73357021 IC50 = 340 nM T62548 CC47ON 76331813 IC50 = 10000 nM T62548 CF9PB2 77105902 IC50 = 70 nM T62548 C5S7CW 86072887 IC50 = 1200 nM T62548 CTW6L4 86072888 IC50 = 160 nM T62548 C0OCM7 86072889 IC50 = 140 nM T62548 CJB2D6 86072906 IC50 = 250 nM T62548 C5CD0N 86072920 IC50 = 300 nM T62548 C1HW4B 89735655 IC50 = 11000 nM T62548 CM0OU7 90472067 IC50 = 316200 nM T62548 CN8V5D 118875292 IC50 = 20000 nM T62548 CPFQ10 118888903 IC50 = 4300 nM T62548 CU2NO8 118888904 IC50 = 130 nM T62548 CHXW78 118888907 IC50 = 1500 nM T62548 CPVX20 118888909 IC50 = 130 nM T62548 CG8IB3 118888910 IC50 = 230 nM T62548 C7L9DW 118888912 IC50 = 60 nM T62548 CH4KC3 118888914 IC50 = 400 nM T62548 CQI01Y 118888915 IC50 > 100000 nM T62548 C6P3LQ 118888916 IC50 = 450 nM T62548 CNH3X7 118888917 IC50 = 690 nM T62548 CW7E1Z 118888918 IC50 = 1900 nM T62548 C2XEP7 118888920 IC50 = 460 nM T62548 CC8U5M 118888921 IC50 = 280 nM T62548 CX9NT0 118888922 IC50 = 680 nM T62548 C5T9WU 118888924 IC50 = 2400 nM T62548 CQP67H 118888925 IC50 = 2000 nM T62548 CT2U0M 118888926 IC50 = 4000 nM T62548 CYN50X 118888927 IC50 = 920 nM T62548 C61BRC 118888929 IC50 = 420 nM T62548 C7CXF9 118888930 IC50 = 14000 nM T62548 CL57HO 118888931 IC50 = 1200 nM T62548 C60FYM 118888932 IC50 = 160 nM T62548 CTP32I 118888933 IC50 = 1200 nM T62548 CTC29U 118888934 IC50 = 250 nM T62548 CU6E8W 118888935 IC50 = 1100 nM T62548 C1TQW8 118888936 IC50 = 44000 nM T62548 CWK0V8 118888937 IC50 = 160 nM T62548 C2QE6K 118888938 IC50 = 4700 nM T62548 C15LEY 118888939 IC50 = 280 nM T62548 CKL47W 118888940 IC50 = 200 nM T62548 CRUI71 118888941 IC50 = 150 nM T62548 CEQ5D3 118888943 IC50 = 460 nM T62548 CW2QI4 127044088 IC50 = 4600 nM T62548 CR8UX2 127044089 IC50 > 100000 nM T62548 CNV07O 130338701 IC50 = 4600 nM T62548 CAOK53 134137419 IC50 = 6300 nM T62548 C06NOP 136227777 IC50 = 6500 nM T62548 C1TY6N 137631658 IC50 = 280 nM T62548 CO0XI5 137632168 IC50 = 170 nM T62548 C8U1CL 137632318 IC50 = 21 nM T62548 CP20NK 137633749 IC50 = 62 nM T62548 CSDJ03 137634374 IC50 = 42 nM T62548 C7F5LK 137634439 EC50 = 930000 nM T62548 CK5LI2 137634643 IC50 = 700 nM T62548 CP6Q3K 137634870 IC50 = 120 nM T62548 C6LQ9T 137634871 IC50 > 10000 nM T62548 C49ENV 137635659 IC50 = 12 nM T62548 CGF95R 137636716 IC50 = 16 nM T62548 C0WQ4T 137637877 IC50 = 290 nM T62548 CXL97Y 137637941 IC50 = 250 nM T62548 C1KP4O 137638201 IC50 = 980 nM T62548 CUIS85 137638312 IC50 = 32 nM T62548 CG2JO7 137638433 IC50 = 1.8 nM T62548 C94BQA 137638520 EC50 = 12000 nM T62548 CXOK62 137639159 IC50 = 44 nM T62548 CS05VB 137639624 IC50 = 130 nM T62548 C8S9CP 137639731 IC50 = 53 nM T62548 C3S2CY 137639895 IC50 = 470 nM T62548 CI0O4Z 137640915 EC50 = 23000 nM T62548 C1SB6C 137642843 IC50 > 10000 nM T62548 C4MQ5Y 137642906 EC50 = 1900000 nM T62548 CPJ26N 137642976 IC50 = 110 nM T62548 CG7Y0B 137644025 IC50 = 560 nM T62548 CS0YG3 137644558 EC50 = 3000 nM T62548 CTF39Y 137644968 IC50 = 140 nM T62548 CVK87P 137645302 IC50 = 200 nM T62548 CV3XS8 137646260 IC50 = 20 nM T62548 C4GH0S 137646432 IC50 = 460 nM T62548 CWQ9E3 137647073 IC50 = 65 nM T62548 C2P6BA 137647099 IC50 = 3800 nM T62548 CX5IK9 137647205 IC50 = 14 nM T62548 C42QMT 137647256 IC50 > 10000 nM T62548 CX5BK1 137647477 EC50 = 87000 nM T62548 CI3F0Q 137647696 IC50 = 17 nM T62548 CJF3E2 137648687 IC50 = 42 nM T62548 C5WL9O 137649838 IC50 = 1700 nM T62548 CK2PS3 137649977 IC50 = 54 nM T62548 C0F3WD 137650435 IC50 = 44 nM T62548 C5OC2K 137650510 EC50 = 120000 nM T62548 C1K7RF 137651597 IC50 = 23 nM T62548 CTE9Q3 137652266 IC50 = 1800 nM T62548 CA46UD 137653406 IC50 = 67 nM T62548 C4OB0A 137653917 IC50 = 370 nM T62548 C7CG5F 137654450 IC50 = 12 nM T62548 C8R0JP 137654554 IC50 = 65 nM T62548 C7NO2X 137654557 IC50 = 3 nM T62548 CQHX89 137654641 IC50 = 100 nM T62548 CGV17I 137654863 EC50 = 220000 nM T62548 CF9H2C 137655150 IC50 > 10000 nM T62548 CSW4Y2 137655245 IC50 = 67 nM T62548 C24DNY 137655381 IC50 = 360 nM T62548 C4W0VL 137656116 IC50 = 7.8 nM T62548 CF0PL4 137656779 IC50 > 10000 nM T62548 CR0QK1 137656838 IC50 = 46 nM T62548 CJ9KZ2 137657230 IC50 = 130 nM T62548 CH08TM 137658866 IC50 = 320 nM T62548 C61FIS 137658873 IC50 = 1200 nM T62548 C5KX6J 137659805 IC50 = 160 nM T62548 CF42ZX 137660643 IC50 = 130 nM T62548 C9T7CJ 137660696 IC50 = 510 nM T62548 CAPY58 137661040 IC50 = 38 nM T62548 CN6QW0 137661458 IC50 = 1100 nM T62548 CFW48S 145967659 IC50 = 1900 nM T62548 CYNP76 145967873 IC50 = 1900 nM T62548 C42CGS 145968147 IC50 = 1600 nM T62548 CGY7E2 145968197 IC50 = 4100 nM T62548 CEM07I 145969035 IC50 = 1400 nM T62548 CUC7I9 145969093 IC50 = 3800 nM T62548 CL1XI2 145969315 IC50 = 640 nM T62548 CJ3VX0 145969342 IC50 = 12000 nM T62548 C3S6TZ 145969486 IC50 = 1500 nM T62548 CK96OA 145969519 IC50 = 540 nM T62548 CTD7P8 145969653 IC50 = 1900 nM T62548 CG4KN3 145969683 IC50 = 500 nM T62548 CEY10F 145970038 IC50 = 29000 nM T62548 CZ96VC 145970244 IC50 = 1800 nM T62548 CM9DW8 145970713 IC50 = 750 nM T62548 CHM13S 145970814 IC50 = 3500 nM T62548 CL9MI5 145970825 IC50 = 430 nM T62548 CE39PX 145970840 IC50 = 200 nM T62548 CI19WX 145970891 IC50 = 340 nM T62548 CC13LU 145970939 IC50 = 830 nM T62548 CXQ19A 145971104 IC50 = 29000 nM T62548 CQJ09K 145986806 IC50 = 2100 nM T62548 C6W9SK 145987049 IC50 = 4100 nM T62548 C2MD1Q 155513187 IC50 > 10000 nM T62548 D04CUA 44256277 IC50 = 460 nM T62548 D0U8UK 11677079 IC50 = 30 nM T75273 D03CQE 5379 IC50 = 287 ug.mL-1 T75273 D0O1WX 2764 IC50 = 4.95 ug.mL-1 T75273 D0VR7W 9571107 IC50 > 200000 nM T75273 D03QAO 25008769 IC50 = 30 nM T75273 D0IY0R 11591505 IC50 = 125 nM T75273 D04OKJ 124093 IC50 > 512 ug.mL-1 T75273 D0T3VO 9865774 IC50 = 7.81 ug.mL-1 T75273 CX9QP0 11837127 IC50 = 27800 nM T75273 C7R6EI 11844920 IC50 = 52300 nM T75273 CY87KS 11997263 IC50 = 21500 nM T75273 CS7JK0 16658873 IC50 = 30 nM T75273 CA9N7S 25022869 IC50 = 3200 nM T75273 C6EJB7 53236573 IC50 = 18700 nM T75273 C61KMA 53236796 IC50 = 12000 nM T75273 CKR1D0 66693299 IC50 > 200000 nM T75273 CI0D9M 73356818 IC50 = 8 nM T75273 CQ7MB8 121415395 IC50 = 1200 nM T75273 C1G2WE 121415404 IC50 = 14000 nM T75273 C5IU4C 121415407 IC50 = 800 nM T75273 C1H8UD 121415415 IC50 = 1100 nM T75273 CG9O1K 121415456 IC50 = 19000 nM T75273 CI51CM 121415469 IC50 = 4500 nM T75273 CB2VC9 121415490 IC50 = 20 nM T75273 CCN1U2 121415509 IC50 = 20 nM T75273 CCT46D 121415540 IC50 < 100 nM T75273 CBL05X 121417642 IC50 = 16900 nM T75273 CE87PY 121417653 IC50 = 164000 nM T75273 CN9T8M 121417654 IC50 = 2100 nM T75273 CZ7XB1 121417677 IC50 = 28300 nM T75273 CSH51T 121417711 IC50 = 20000 nM T75273 C2IRX6 121417737 IC50 > 100000 nM T75273 C6OP3Z 121418109 IC50 = 12100 nM T75273 CH08PV 121429867 IC50 = 2800 nM T75273 C3FW9K 121433130 IC50 = 10500 nM T75273 CAT23Q 132961614 IC50 = 0.214 ug.mL-1 T75273 CL2WR6 132961615 IC50 = 0.357 ug.mL-1 T75273 C76UHD 132961616 IC50 = 0.328 ug.mL-1 T75273 CSL5J8 132961617 IC50 = 0.214 ug.mL-1 T75273 CCD5K9 134129921 IC50 = 0.214 ug.mL-1 T75273 C8XYI7 134130806 IC50 = 0.214 ug.mL-1 T75273 CWT8L1 134149458 IC50 = 0.214 ug.mL-1 T75273 C9HO5W 134156187 IC50 = 0.214 ug.mL-1 T75273 C9QH8D 142332183 IC50 = 25.1 ug.mL-1 T75273 C1E6LY 145950292 IC50 = 5.11 ug.mL-1 T75273 C5PR8D 145951648 IC50 = 0.71 ug.mL-1 T75273 CUJ0T9 145953207 IC50 = 2.11 ug.mL-1 T75273 C0I1HC 145957648 IC50 = 2.69 ug.mL-1 T75273 CY6C0S 145972903 IC50 = 0.79 ug.mL-1 T75273 C57TMP 155511431 IC50 = 43300 nM T75273 CUZ0M6 155522161 IC50 = 26800 nM T75273 CAJ91F 155531127 IC50 = 1600 nM T75273 C09COM 155532384 IC50 = 3900 nM T75273 C4V7UR 155538148 IC50 = 7800 nM T75273 CXJ1G9 155544331 IC50 = 9600 nM T75273 C7UDQ2 155545881 IC50 = 600 nM T75273 CLB2V4 155546018 IC50 = 33100 nM T75273 C79USC 155548113 IC50 = 1500 nM T75273 CG4E8A 155548135 IC50 = 2600 nM T75273 CED32V 155549037 IC50 = 12100 nM T75273 CIR6C4 155549058 IC50 = 3700 nM T75273 CQ7T6H 155549145 IC50 = 6900 nM T75273 C06ZCE 155556229 IC50 = 6800 nM T75273 CZUE35 155558181 IC50 = 5200 nM T75273 CIW64O 155560768 IC50 = 1100 nM T75273 CXW42N 155563849 IC50 = 1300 nM T75273 C9E5MU 155566312 IC50 = 4600 nM T75273 CQYI40 155568240 IC50 = 3600 nM T75273 D05LOY 16048804 IC50 = 4200 nM T75273 D0C9BH 54706138 IC50 = 0.648 ug.mL-1 T10670 D0LI1C 44469321 IC50 > 10000 nM T10670 D0V2GT 5311023 Ki > 10000 nM T10670 C9NG4X 16033 EC50 = 0.0631 nM T10670 C74KDN 624746 IC50 > 10000 nM T10670 C1Q4WZ 1294837 Ki = 501.19 nM T10670 C1AI0D 2223246 IC50 = 440 nM T10670 C51PSM 2936384 IC50 = 190 nM T10670 CP8NR5 2936750 IC50 = 1100 nM T10670 CVKX10 2945439 IC50 = 207 nM T10670 C4SO3U 3236979 IC50 = 1200 nM T10670 C7CNR4 4268834 IC50 = 371 nM T10670 CDO51W 4460128 IC50 = 4400 nM T10670 CF20QJ 4527770 Ki > 31622.78 nM T10670 C39UDN 5312114 IC50 = 1890 nM T10670 C2T3BN 6011884 IC50 = 4000 nM T10670 CI26VT 9799669 IC50 > 30000 nM T10670 C5MC8Y 9802119 IC50 > 10000 nM T10670 CK7QY8 9867212 IC50 > 30000 nM T10670 CT7S5I 9869041 IC50 > 10000 nM T10670 CPGD84 9887225 IC50 > 10000 nM T10670 CS92LR 9916525 Ki > 10000 nM T10670 CWP3V6 9930778 IC50 >> 1000 nM T10670 C7N5SJ 10003722 IC50 > 10000 nM T10670 CH1Q6E 10008757 Ki > 3000 nM T10670 CK3W5X 10030299 Ki > 3000 nM T10670 C73QBA 10047509 IC50 > 10000 nM T10670 CL96TH 10110741 IC50 > 10000 nM T10670 C6IXU4 10293988 Ki > 10000 nM T10670 C8L7WY 10295464 IC50 > 30000 nM T10670 CX2W6U 10323693 IC50 = 600 nM T10670 CCOY30 10369730 IC50 = 350 nM T10670 CA1C6E 10418848 Ki = 11.3 nM T10670 C4HMY5 10429613 IC50 = 2682 nM T10670 C5IW8S 10456979 IC50 = 450 nM T10670 C84MSG 10524003 Ki > 10000 nM T10670 CKQ2G1 10531484 Ki > 10000 nM T10670 CQ1P5I 10554658 Ki > 10000 nM T10670 C0F9SD 10555187 Ki > 10000 nM T10670 C0FP2G 10619067 Ki > 10000 nM T10670 CZ0U1P 10625004 Ki > 10000 nM T10670 C3L6TA 10671331 Ki > 10000 nM T10670 C7MC2O 10672357 Ki > 10000 nM T10670 C6HQ1X 10692519 Ki > 10000 nM T10670 CS4JF0 10820168 Ki = 1650 nM T10670 CEH6O1 10820196 Ki = 1420 nM T10670 CGT23W 10872843 IC50 > 10000 nM T10670 CFHD79 10915843 IC50 > 10000 nM T10670 CDMB60 10916418 IC50 = 1101 nM T10670 C21PAY 10927348 IC50 > 10000 nM T10670 CJ0OF1 10949261 IC50 > 10000 nM T10670 CM54HE 10959710 IC50 > 10000 nM T10670 C08VWM 10971892 IC50 > 10000 nM T10670 CO98AV 10982716 IC50 > 10000 nM T10670 CI6W3N 10993145 IC50 > 10000 nM T10670 CGSF91 11013840 IC50 > 10000 nM T10670 C1ICL8 11025578 IC50 > 10000 nM T10670 C4UPT2 11057893 IC50 > 10000 nM T10670 CKC6D3 11133371 IC50 > 10000 nM T10670 CL9G0U 11156574 IC50 = 15000 nM T10670 C1GRD9 11165586 IC50 = 30000 nM T10670 CK0RO5 11179227 IC50 = 800 nM T10670 C2EX7A 11192050 IC50 = 8900 nM T10670 CKMQ07 11203099 IC50 = 2500 nM T10670 CGV85T 11203422 IC50 = 1100 nM T10670 C16ZKM 11214627 IC50 = 1900 nM T10670 CS8RO0 11225709 IC50 = 30000 nM T10670 CT0I2W 11236647 IC50 = 3500 nM T10670 C1XRS4 11236982 IC50 = 12000 nM T10670 CKX8M5 11237245 IC50 = 12000 nM T10670 C4N1AS 11249185 IC50 = 3900 nM T10670 C8UQ6A 11261330 IC50 = 30000 nM T10670 CKHY73 11271868 IC50 = 26000 nM T10670 CKX43W 11272082 IC50 = 1000 nM T10670 CXLZ69 11294247 IC50 = 17500 nM T10670 CU95IG 11294696 IC50 = 3200 nM T10670 C5T1JZ 11295383 IC50 = 4800 nM T10670 C2N9WX 11306287 IC50 = 1100 nM T10670 C0ATK7 11306461 IC50 = 29000 nM T10670 C64UBZ 11307880 IC50 = 5800 nM T10670 CSV26Z 11316909 IC50 = 5300 nM T10670 C23CUQ 11318105 IC50 = 2800 nM T10670 CEC8I7 11318800 IC50 = 2800 nM T10670 C8XE2M 11328497 IC50 = 12000 nM T10670 C03TDS 11330404 IC50 = 3300 nM T10670 CXO5V9 11340260 IC50 = 30000 nM T10670 CB1M0V 11353113 IC50 = 30000 nM T10670 CI0CV3 11364830 IC50 = 30000 nM T10670 CE6W7N 11375032 IC50 = 16000 nM T10670 C2PTX9 11375033 IC50 = 22000 nM T10670 C9H7TX 11375413 IC50 = 3600 nM T10670 CS84JE 11387103 IC50 = 4800 nM T10670 C1PA4G 11397239 IC50 = 17000 nM T10670 CJ6A5V 11398198 IC50 = 30000 nM T10670 C34TMN 11408945 IC50 = 30000 nM T10670 CGE85F 11409805 IC50 = 1100 nM T10670 C85LYP 11430418 IC50 > 1000 nM T10670 CZ7XC9 11431881 IC50 = 10000 nM T10670 C6EFU2 11443018 IC50 = 30000 nM T10670 CM65FB 11453411 IC50 = 22000 nM T10670 C6E5RQ 11453755 IC50 = 30000 nM T10670 C5C4EA 11454489 IC50 = 18000 nM T10670 CGZ2T7 11465776 IC50 = 30000 nM T10670 C7RFS3 11466430 IC50 = 3000 nM T10670 CB1U2O 11477689 IC50 = 2300 nM T10670 CK2Q9F 11478324 IC50 = 500 nM T10670 C79VWO 11489162 IC50 = 3600 nM T10670 CQ49SB 11640844 Ki > 10000 nM T10670 C1YWG5 11732188 IC50 > 10000 nM T10670 CX1H9T 11751925 IC50 = 9200 nM T10670 CZSR54 11752266 IC50 = 1400 nM T10670 C43LHB 11760541 IC50 > 10000 nM T10670 CJ5TE0 11798404 Ki > 10000 nM T10670 CUM43R 12071667 IC50 > 10000 nM T10670 CTYR34 16058735 IC50 = 15 nM T10670 CFAG02 16665228 IC50 = 20 nM T10670 CL50QA 16666511 IC50 = 50 nM T10670 CAW9R5 16666777 IC50 = 530 nM T10670 CLUZ85 16667089 IC50 = 370 nM T10670 CCEJ98 16667090 IC50 = 12 nM T10670 CFH87Q 16667091 IC50 = 12 nM T10670 CU4IW5 16667135 IC50 = 37 nM T10670 CWV95M 16667180 IC50 = 16 nM T10670 COR4A5 16667181 IC50 = 20 nM T10670 CCMO72 16667279 IC50 = 33 nM T10670 CX2P8T 16667331 IC50 = 165 nM T10670 CF0S5Q 17118052 Ki = 6.31 nM T10670 CO5PA8 17312686 IC50 = 178 nM T10670 C8WK1T 17376722 IC50 = 8162 nM T10670 CIYU59 20587808 IC50 > 10000 nM T10670 C7CGH0 20773956 IC50 = 220 nM T10670 CHMZ61 20773958 IC50 = 240 nM T10670 C4Q8KN 21129772 IC50 > 100000 nM T10670 CEOA23 22254020 IC50 > 1000 nM T10670 CBS20U 22254050 IC50 > 1000 nM T10670 CO32YX 22254068 IC50 > 1000 nM T10670 CHQT84 22254131 IC50 > 1000 nM T10670 CP7E2N 22325336 IC50 > 10000 nM T10670 CC2WI6 22499399 IC50 = 530 nM T10670 CFJ7W3 22779969 Ki = 79.43 nM T10670 CG3VL7 25067562 IC50 > 10000 nM T10670 CY2R4C 25134625 IC50 = 6 nM T10670 C50SQO 25151875 IC50 = 14 nM T10670 C7YAZ6 25151876 IC50 = 9 nM T10670 CIJ58E 25151877 IC50 = 42 nM T10670 C7IH3J 25181112 Ki > 10000 nM T10670 C7VID1 25211875 IC50 > 10000 nM T10670 CSHE98 42628839 IC50 = 11 nM T10670 C89WIH 42628851 IC50 = 7 nM T10670 CNU7P4 42630820 IC50 > 10000 nM T10670 CF1C8G 42643943 IC50 = 740 nM T10670 C7QL2U 42644181 IC50 = 420 nM T10670 CZ7B3I 42647046 IC50 = 240 nM T10670 CTY7N2 42647272 IC50 = 220 nM T10670 CZI94L 42647273 IC50 = 10000 nM T10670 CHG3D4 44128297 IC50 = 34 nM T10670 CLX51J 44249749 Ki = 25.12 nM T10670 CJ1VA7 44274435 IC50 = 11000 nM T10670 CH3A4G 44274493 IC50 = 17000 nM T10670 C6KR1Y 44287938 IC50 = 78000 nM T10670 CHT17W 44287971 IC50 = 540000 nM T10670 C2IXS5 44287982 IC50 > 400000 nM T10670 C7X5DG 44287999 IC50 = 177000 nM T10670 C1FW4N 44288067 IC50 = 247000 nM T10670 CAI9T7 44288112 IC50 = 575000 nM T10670 CN76WT 44288390 IC50 = 97000 nM T10670 CS1FG8 44288395 IC50 = 59000 nM T10670 CH0U3I 44329247 IC50 = 10000 nM T10670 CK0EX9 44329354 IC50 = 1000 nM T10670 C2F6IE 44329355 IC50 > 10000 nM T10670 CT14FA 44329364 IC50 > 10000 nM T10670 C5SGW2 44329380 IC50 > 10000 nM T10670 CDPA43 44329396 IC50 = 3700 nM T10670 C8MC6O 44329420 IC50 > 10000 nM T10670 C97BSL 44329428 IC50 = 2200 nM T10670 CAO5Q6 44329441 IC50 > 10000 nM T10670 CJ0SF8 44329449 IC50 > 10000 nM T10670 CD2M6Z 44329450 IC50 = 450 nM T10670 CYA91D 44329467 IC50 > 10000 nM T10670 C5V0ET 44342972 IC50 = 0.39 nM T10670 CTX16Q 44351135 Ki = 2.5 nM T10670 C1NUA7 44351136 Ki = 0.6 nM T10670 CD87HA 44351182 Ki = 0.4 nM T10670 CNOB51 44351197 Ki = 1.3 nM T10670 CJM96N 44461116 IC50 > 30000 nM T10670 C4DL5C 44469677 IC50 > 10000 nM T10670 C68NXC 44517723 IC50 = 1400 nM T10670 CZ65XF 44579887 IC50 > 10000 nM T10670 CVO10S 44580050 IC50 > 10000 nM T10670 C61HUP 45267282 Ki = 316.23 nM T10670 CCV95O 45267291 Ki > 6309.57 nM T10670 C5KUT9 45268145 Ki = 199.53 nM T10670 C8QKO0 45268150 Ki = 158.49 nM T10670 CA9LK6 45268152 Ki = 19.95 nM T10670 C1F9WM 45268155 Ki = 316.23 nM T10670 C4UXF7 45268161 Ki = 63.1 nM T10670 CG2R4Q 45269027 Ki = 50.12 nM T10670 CE1MT9 45269036 Ki = 316.23 nM T10670 CF7V3A 45269040 Ki = 316.23 nM T10670 C0QVA8 45269874 Ki = 79.43 nM T10670 C6DE1V 45269879 Ki = 2511.89 nM T10670 CK0VC1 45269889 Ki = 10 nM T10670 CM3SG6 45269896 Ki = 3162.28 nM T10670 C1T2AU 45269902 Ki = 2.512 nM T10670 C65RMJ 45271522 Ki = 125.89 nM T10670 C90NSE 45271528 Ki = 158.49 nM T10670 CFC28M 45271536 Ki = 5.012 nM T10670 C65BQL 45271540 Ki = 1584.89 nM T10670 CEL01G 45271544 Ki = 12.59 nM T10670 C8P9BT 45272450 Ki = 630.96 nM T10670 C94KLT 45272453 Ki = 3.981 nM T10670 C9FCB4 45273317 Ki = 12.59 nM T10670 CA1ET4 45273325 Ki = 2511.89 nM T10670 C30LDO 45487447 IC50 > 10000 nM T10670 CL9PW1 45487448 IC50 > 10000 nM T10670 C5YB1P 46231125 Ki = 11.3 nM T10670 CZD7T5 46880224 Ki > 10000 nM T10670 CGO62F 50925473 Ki = 158.49 nM T10670 CTF13N 50925474 Ki = 125.89 nM T10670 C07UHK 50925475 Ki = 25.12 nM T10670 C1X2NF 50925491 Ki = 19.95 nM T10670 CY28CM 50925492 Ki = 1.995 nM T10670 CC7TM4 52941248 Ki = 398.11 nM T10670 CAF49Q 52942479 Ki = 50.12 nM T10670 CPT97A 52942508 Ki = 251.19 nM T10670 CZ1XW7 52943629 Ki = 251.19 nM T10670 CFJ40D 52943733 Ki = 794.33 nM T10670 CXK83V 52945324 Ki = 316.23 nM T10670 CPB2Q6 52946124 Ki = 1995.26 nM T10670 C6D5RE 52946147 Ki = 1258.93 nM T10670 CS50AK 52947300 Ki = 316.23 nM T10670 C0E1XO 52947327 Ki = 251.19 nM T10670 C7CU2P 52947370 Ki = 1000 nM T10670 C8NL5G 52947375 Ki = 79.43 nM T10670 CST85B 52947384 Ki = 398.11 nM T10670 CV6CQ3 52948513 Ki = 125.89 nM T10670 C4SV8W 52948566 Ki = 63.1 nM T10670 C01PRX 52948640 Ki = 15.85 nM T10670 C1U7YB 52948948 Ki = 15.85 nM T10670 C10JNO 52949765 Ki = 199.53 nM T10670 CP84KG 52949775 Ki = 199.53 nM T10670 C4U6OX 52949776 Ki = 79.43 nM T10670 CY9QM5 52949834 Ki = 630.96 nM T10670 CQ18SU 52950120 Ki = 501.19 nM T10670 CH5A3Z 52953217 Ki > 3000 nM T10670 CV10HR 52953219 Ki > 500 nM T10670 C3M2KC 56659929 IC50 = 25 nM T10670 CZCT67 56659930 IC50 = 35 nM T10670 CWD1Y2 56659931 IC50 = 11 nM T10670 CQ4V5H 56659932 IC50 = 30 nM T10670 CX2MI3 56670258 IC50 = 37 nM T10670 CC81DQ 56670259 IC50 = 40 nM T10670 CX9F1G 56670260 IC50 = 10 nM T10670 C74QMI 56672399 IC50 = 200 nM T10670 CI37FT 56673774 IC50 = 52 nM T10670 CYRA39 56673775 IC50 = 25 nM T10670 CYF2A0 56677101 IC50 = 100 nM T10670 CQ75OA 56680424 IC50 = 150 nM T10670 CO37WR 56680425 IC50 = 37 nM T10670 CLQ9Y2 56841989 Ki = 0.25 nM T10670 C7ARQ6 58055717 IC50 = 600 nM T10670 CH02MJ 58055719 IC50 = 830 nM T10670 CUL3I4 58055738 IC50 = 480 nM T10670 C38PGB 58055741 IC50 = 85 nM T10670 C3J7DE 58055745 IC50 = 78 nM T10670 C0F3YZ 58055750 IC50 = 810 nM T10670 CM4YI1 58055756 IC50 = 110 nM T10670 CX0DB5 58055758 IC50 = 41 nM T10670 C48GAX 58055759 IC50 = 270 nM T10670 CHRJ92 58055769 IC50 = 1950 nM T10670 C62TIB 58055771 IC50 = 130 nM T10670 CDF51E 58055778 IC50 = 900 nM T10670 CAOZ08 58055782 IC50 = 160 nM T10670 CU9QA7 58055783 IC50 = 460 nM T10670 CQN58S 58870638 IC50 = 25 nM T10670 C1YCO9 58870642 IC50 = 26 nM T10670 CQK1J7 58870644 IC50 = 70 nM T10670 C9B2MX 58870648 IC50 = 3000 nM T10670 C7F8XA 58870651 IC50 = 40 nM T10670 C8O0XY 58870667 IC50 = 100 nM T10670 C98APS 58870679 IC50 = 200 nM T10670 CZMF59 58870680 IC50 = 100 nM T10670 CE5WK7 58870701 IC50 = 80 nM T10670 CHXU89 58870727 IC50 = 300 nM T10670 CRA92I 58870729 IC50 = 26 nM T10670 CCN2O0 58870731 IC50 = 44 nM T10670 CGO5R7 58870735 IC50 = 162 nM T10670 CWE6V8 58870752 IC50 = 14 nM T10670 C4BLE2 58870759 IC50 = 70 nM T10670 CG8BU0 58870763 IC50 = 330 nM T10670 C38WGO 58870766 IC50 = 65 nM T10670 C32LPR 58870776 IC50 = 150 nM T10670 CX0C2L 58870783 IC50 = 72 nM T10670 C5NG4E 58870814 IC50 = 18 nM T10670 CD0FN8 58870834 IC50 = 50 nM T10670 CW0CR2 66561564 IC50 = 19 nM T10670 CR9QG5 66561565 IC50 = 12 nM T10670 C70DBL 67678347 IC50 = 170 nM T10670 CW68SD 68872605 IC50 = 290 nM T10670 C6AT2F 68873961 IC50 = 150 nM T10670 C2R1EC 69089436 IC50 = 38 nM T10670 CV73UG 69305104 IC50 = 44 nM T10670 CL6R8B 69669928 IC50 = 33 nM T10670 COB41D 69670041 IC50 = 240 nM T10670 CDC58E 69670197 IC50 = 27 nM T10670 CZL6E8 69670211 IC50 = 27 nM T10670 C65XGC 69670294 IC50 = 720 nM T10670 CB24DP 70681544 IC50 = 777 nM T10670 C2YA5S 70681545 IC50 = 301 nM T10670 C6KD9T 70681546 IC50 = 136 nM T10670 CC8Q0N 70681549 IC50 > 10000 nM T10670 CWY8V2 70681551 IC50 = 483 nM T10670 C8I0GP 70681552 IC50 = 248 nM T10670 CO46GT 70683658 IC50 = 1200 nM T10670 C9QNK8 70683659 IC50 = 271 nM T10670 CY7X1Z 70683661 IC50 = 6760 nM T10670 CPH2W4 70683662 IC50 = 1580 nM T10670 C6QAS0 70683663 IC50 = 59 nM T10670 CQW93J 70685785 IC50 = 1770 nM T10670 C1RK3Q 70685805 IC50 = 899 nM T10670 CZSE08 70685806 IC50 = 1350 nM T10670 CK6IS7 70685808 IC50 = 89 nM T10670 CWP73D 70687925 IC50 = 121 nM T10670 CB3RO4 70687926 IC50 = 238 nM T10670 CP52BA 70687927 IC50 = 98 nM T10670 C4HY2W 70687928 IC50 = 2680 nM T10670 CM4QP1 70687929 IC50 = 220 nM T10670 CYSA03 70689958 IC50 = 612 nM T10670 CLK0X7 70689959 IC50 = 72 nM T10670 C5VSD0 70689960 IC50 = 78 nM T10670 CZB3G6 70689961 IC50 = 323 nM T10670 CO5C0L 70689962 IC50 = 3300 nM T10670 C7MNV6 70689963 IC50 = 49 nM T10670 C8Y3VE 70689965 IC50 = 394 nM T10670 C83EWV 70692113 IC50 = 141 nM T10670 CIG05H 70694148 IC50 = 1047 nM T10670 C2DHG4 70696286 IC50 = 1419 nM T10670 CM28SQ 70696287 IC50 = 206 nM T10670 C5J9CW 70696288 IC50 = 117 nM T10670 CJY5O0 70696289 IC50 = 6079 nM T10670 CY74MW 70696290 IC50 = 85 nM T10670 C9IUC7 70696292 IC50 = 67 nM T10670 C2QS4L 70696293 IC50 = 61 nM T10670 CM2S5E 71574720 Ki = 9.9 nM T10670 CZ6N5M 71713624 IC50 = 45 nM T10670 CC9S1T 71713780 IC50 = 12 nM T10670 CM09QV 71713781 IC50 = 24 nM T10670 C8XR4A 71713782 IC50 = 70 nM T10670 C3BR8Z 71713783 IC50 = 665 nM T10670 CYLM84 71713784 IC50 = 476 nM T10670 CQS27Y 71713934 IC50 = 7 nM T10670 C21QNH 71713935 IC50 = 27 nM T10670 CGKU71 71717895 Ki = 0.7 nM T10670 C8QO1W 71719108 Ki = 2.6 nM T10670 C9UH7J 72205287 Ki > 5000 nM T10670 CA26US 72205877 Ki > 5000 nM T10670 CWH6T3 72548703 IC50 = 0.28 nM T10670 CFV1X0 72711815 Ki > 1000 nM T10670 CE6KV1 72712030 Ki > 1000 nM T10670 CFQY96 73345485 Ki = 1.5 nM T10670 C1X2AR 73346549 Ki > 5000 nM T10670 CJ5HR8 73347019 Ki = 2.3 nM T10670 CPXJ28 73349570 Ki > 5000 nM T10670 C1NQ7B 73350103 Ki = 0.3 nM T10670 CTJ3D0 73350105 Ki = 1.1 nM T10670 C0NM1P 73351119 Ki > 1000 nM T10670 CB9R8P 73353058 Ki = 0.3 nM T10670 CO4GL8 73353059 Ki = 0.3 nM T10670 CRC73X 73354075 Ki > 1000 nM T10670 CRL10F 73354088 Ki > 5000 nM T10670 CIFL82 73354092 Ki > 5000 nM T10670 C9XCU8 73354094 Ki > 5000 nM T10670 C34SQD 73354098 Ki = 7 nM T10670 CCK72G 73355613 Ki > 5000 nM T10670 CO26NJ 73355617 Ki = 620 nM T10670 CUM6D5 73357147 Ki > 1000 nM T10670 CVR97L 76313843 IC50 = 9200 nM T10670 C6N1HQ 76321090 IC50 = 340 nM T10670 CZR0V5 76321091 IC50 = 35 nM T10670 CK29MI 76321092 IC50 = 11000 nM T10670 CMF5J8 76324740 IC50 = 3700 nM T10670 CPSF81 76324741 IC50 = 22000 nM T10670 CGU64Q 76328289 IC50 = 300 nM T10670 C8QJW0 76335552 IC50 = 30000 nM T10670 CB3FG4 85472343 Ki = 950 nM T10670 C8N1LM 87725189 EC50 = 0.2 nM T10670 CK5B7R 118718116 Ki = 0.2 nM T10670 C94LWU 118718124 Ki = 2.2 nM T10670 CJ5Q9R 118718125 Ki = 1 nM T10670 C92ZVT 118718320 Ki = 3.6 nM T10670 CT5QV3 122178178 EC50 > 1000 nM T10670 CK3W1J 122178179 EC50 > 1000 nM T10670 CJ3YC7 122178180 EC50 > 1000 nM T10670 CDB67H 122178181 EC50 = 0.6 nM T10670 C0DKP8 122178182 EC50 = 0.5 nM T10670 CLZ87K 122178183 EC50 = 0.3981 nM T10670 C3LKE9 122178186 EC50 = 1.585 nM T10670 CE0WR2 122178187 EC50 = 3.9 nM T10670 C4XDU8 122178188 EC50 = 3.162 nM T10670 C5Q7WR 122178189 EC50 = 1.995 nM T10670 CW2BG8 127029975 Ki = 1700 nM T10670 C7Q2WP 127030359 Ki = 1300 nM T10670 CK0A1M 127031281 Ki = 730 nM T10670 C0XR6M 127041306 Ki > 3000 nM T10670 C5PA2G 127041908 Ki > 10000 nM T10670 C7TM1Y 127042243 Ki > 10000 nM T10670 C62JIE 127042244 Ki > 3000 nM T10670 CA1ZE0 137632397 EC50 = 0.21 nM T10670 C24XZR 137632601 EC50 = 4.4 nM T10670 CF43NZ 137634023 EC50 = 0.16 nM T10670 CKD7R2 137634108 EC50 = 1.8 nM T10670 C2B9HY 137634335 EC50 = 3.8 nM T10670 CQ2P4C 137634780 EC50 = 0.74 nM T10670 CTF21Z 137635521 EC50 = 4.6 nM T10670 C3SH2T 137635909 EC50 = 4.6 nM T10670 CW9FB2 137636973 EC50 = 1.7 nM T10670 CMU05F 137637360 EC50 = 0.2 nM T10670 CG8R9K 137637445 EC50 = 2.5 nM T10670 C5ULH2 137637657 EC50 = 0.2 nM T10670 CO9T3A 137638459 EC50 = 0.28 nM T10670 C4TRA5 137638723 EC50 = 0.61 nM T10670 C7DY9P 137639373 EC50 = 0.19 nM T10670 CR47GV 137639719 EC50 = 1 nM T10670 CNHO10 137639723 EC50 = 2 nM T10670 CU3G2O 137640909 EC50 = 1.3 nM T10670 CZ0N6M 137641708 EC50 = 0.068 nM T10670 C0CFJ9 137641883 EC50 = 4.2 nM T10670 CJBS04 137641937 EC50 = 0.48 nM T10670 CFPM41 137642856 EC50 = 2.5 nM T10670 C4RZQ2 137643080 EC50 = 0.61 nM T10670 CHBE91 137643148 EC50 = 1.3 nM T10670 CTNG60 137644502 EC50 = 0.33 nM T10670 CCXK08 137646370 EC50 = 0.41 nM T10670 C12KSF 137646917 EC50 = 1.2 nM T10670 C6K1WR 137648110 EC50 = 5.5 nM T10670 C14XTE 137649292 EC50 = 6.4 nM T10670 CY6SU8 137649686 EC50 = 0.75 nM T10670 CF84XP 137650904 EC50 = 3 nM T10670 C4A6GP 137651435 EC50 = 3.8 nM T10670 CA2D0K 137651823 EC50 = 0.2 nM T10670 CY7XR8 137653207 EC50 = 0.55 nM T10670 C4E8CB 137655430 EC50 = 0.2 nM T10670 C9B3IS 137657064 EC50 = 1 nM T10670 CD26FG 137658962 EC50 = 0.42 nM T10670 CYFM76 137659071 EC50 = 0.59 nM T10670 C2EI8S 137660151 EC50 = 2 nM T10670 C0P9LD 137660673 EC50 = 0.6 nM T10670 C42WVE 137661485 EC50 = 0.66 nM T10670 C3YB4L 145965033 EC50 = 0.13 nM T10670 CX3N0D 145965127 EC50 = 0.41 nM T10670 C80DTH 145965778 EC50 = 0.35 nM T10670 CG8SN7 145965939 EC50 = 0.15 nM T10670 CYGH78 145966137 EC50 = 0.49 nM T10670 CGU81X 145967047 EC50 = 0.17 nM T10670 C3QWV8 145967161 EC50 = 0.8 nM T10670 C5J8PT 145967318 EC50 = 0.5 nM T10670 C3BW8K 145967399 EC50 = 0.28 nM T10670 CYPL17 145967423 EC50 = 0.13 nM T10670 C3EB6F 145967575 IC50 = 13 nM T10670 CZ0DU2 145967577 IC50 = 7.6 nM T10670 C7W4AV 145968270 IC50 = 24 nM T10670 CJ52UG 145969510 IC50 = 3.4 nM T10670 CX8AB1 145969670 IC50 = 13 nM T10670 CUDL74 145969969 IC50 = 7.6 nM T10670 CBS06Y 145970108 IC50 = 0.19 nM T10670 C1O2UV 145970168 IC50 = 0.19 nM T10670 C7R0VW 145970558 IC50 = 4.5 nM T10670 COIX85 145971139 IC50 = 8 nM T10670 CY73PI 145972295 EC50 = 0.4 nM T10670 CZAC30 145972608 EC50 = 0.17 nM T10670 CW17FS 145973526 EC50 = 0.14 nM T10670 C1MKR3 145973561 EC50 = 0.28 nM T10670 CM19IH 145974475 EC50 = 0.5 nM T10670 C0QFU2 145976002 EC50 = 0.16 nM T10670 CD0C6A 145976367 EC50 = 0.21 nM T10670 CJ69CO 145976419 EC50 = 0.11 nM T10670 C4U9EI 145977518 EC50 = 0.59 nM T10670 C2OEC4 145977697 EC50 = 0.18 nM T10670 CP6ZH4 145977725 EC50 = 0.11 nM T10670 CLI06K 145977835 EC50 = 0.18 nM T10670 CH0RS5 145978112 EC50 = 0.17 nM T10670 CC0YM4 145978304 EC50 = 2 nM T10670 CH8BD7 145978818 EC50 = 0.13 nM T10670 C97IBF 145978857 EC50 = 0.21 nM T10670 C8ZAN2 145979152 Ki = 6.3 nM T10670 C4SB9P 145979291 Ki = 3.1 nM T10670 CQ78WY 145979469 Ki = 250 nM T10670 CO1M3D 145979616 Ki = 79 nM T10670 C3OXL9 145979975 Ki = 2500 nM T10670 C4H9BZ 145980763 Ki = 0.25 nM T10670 CH5MZ8 145980782 Ki = 1.259 nM T10670 CI5F7E 145980802 Ki = 1258.93 nM T10670 CP4RI5 145980997 Ki = 1.259 nM T10670 CW80EN 145981168 Ki = 1584.89 nM T10670 CTF1C6 145981319 Ki = 7900 nM T10670 COB75I 145981742 Ki = 1.995 nM T10670 C60AUT 145981829 Ki = 1.995 nM T10670 COF9U8 145982156 Ki = 50 nM T10670 CXE2K1 145984150 Ki = 0.79 nM T10670 CM4VG2 145984378 Ki = 0.5 nM T10670 CG74XB 145985156 Ki = 39.81 nM T10670 C5XL9U 145985176 EC50 > 30 nM T10670 C63DRI 145985639 Ki = 79 nM T10670 C5UDH2 145986414 Ki = 199.53 nM T10670 CLEQ40 145986472 Ki = 0.3981 nM T10670 CZ68SU 145986539 Ki = 1995.26 nM T10670 CGB4Y3 145987289 Ki = 158.49 nM T10670 CI1XY0 145987577 Ki = 630 nM T10670 C4T5IJ 145987618 Ki = 1000 nM T10670 CL2I3Y 145987802 Ki = 1000 nM T10670 CIZ94Y 145988210 Ki = 316.23 nM T10670 CRW15D 145989250 Ki = 25 nM T10670 C5O8AZ 145989327 Ki = 0.63 nM T10670 CG63IW 145989789 Ki = 158.49 nM T10670 CF5OV2 145990257 Ki = 2.5 nM T10670 CH50MF 145991293 Ki = 2.5 nM T10670 CDX86E 145991438 Ki = 39.81 nM T10670 C6PS8F 145991876 Ki = 6.3 nM T10670 C7K8CT 145992181 Ki = 0.79 nM T10670 CC72HP 145992661 Ki = 5 nM T10670 C5KF0O 145992989 Ki = 250 nM T10670 CQH29C 145993358 Ki = 1584.89 nM T10670 C9Z4PM 145993376 Ki = 50 nM T10670 CAZ6I7 145993698 Ki = 2.5 nM T10670 CPD7M9 145994220 Ki = 1.259 nM T10670 CQF01J 155524657 Ki = 830 nM T10670 CCK32B 155543070 Ki = 420 nM T10670 CCZ09U 155547323 Ki > 3000 nM T10670 C1T7DH 155549336 Ki = 750 nM T10670 CDT81L 155553742 Ki > 10000 nM T10670 CX43VE 155561277 Ki > 10000 nM T10670 C4M9NL 155561620 Ki > 3000 nM T10670 D00OLA 44409453 Ki = 50 nM T10670 D02WBY 10324083 IC50 = 63.1 nM T10670 D07OOG 73347134 Ki = 390 nM T10670 D08YWE 73348635 Ki = 260 nM T10670 D0G4HT 73354703 Ki = 890 nM T10670 D0J9VA 44409452 Ki = 1050 nM T10670 D0Q2IU 44439563 EC50 = 430 nM T10670 D0V0HM 73345612 Ki = 360 nM T02703 D08ZEB 2733 IC50 = 14100 nM T02703 D05QJT 9797017 IC50 = 70 nM T02703 D0D3AI 39836 IC50 = 8000 nM T02703 D0V0NL 2146 IC50 = 3900 nM T02703 D0R5XK 9815538 Ki = 1.8 nM T02703 D0Y7VJ 2733506 IC50 = 100 nM T02703 CHM9K2 4366 IC50 = 340 nM T02703 C9OF8C 5142 IC50 = 3000 nM T02703 C3W0JR 11379 IC50 = 1700 nM T02703 C20EWK 15347 IC50 = 940 nM T02703 CL81BQ 15348 IC50 = 600 nM T02703 C6WDC5 15765 IC50 = 2000 nM T02703 C5TXR9 27842 IC50 = 800 nM T02703 C9NY7L 73046 IC50 = 1800 nM T02703 C8CQW2 73742 IC50 = 4600 nM T02703 CN18AG 83053 IC50 = 790 nM T02703 C7AB0Y 107968 IC50 = 300 nM T02703 CZXU91 118425 IC50 = 1100 nM T02703 CQ3RW8 124357 Ki = 2200 nM T02703 CP49UZ 132862 IC50 = 300 nM T02703 CT7M5K 135193 IC50 = 830 nM T02703 CWG0F1 152144 IC50 = 1500 nM T02703 CW72NB 203391 Ki > 50000 nM T02703 CG96BR 211124 IC50 > 50000 nM T02703 C23ABJ 262484 IC50 = 7200 nM T02703 C8B7YF 287208 IC50 > 50000 nM T02703 CJ0T9Y 311869 IC50 > 50000 nM T02703 CC1X3J 317495 IC50 = 59 nM T02703 C3ZA0H 322632 IC50 = 9900 nM T02703 CV7K2N 322634 IC50 > 50000 nM T02703 CTK6I8 330841 IC50 = 3200 nM T02703 C41OMP 430989 IC50 = 25000 nM T02703 CK9U6L 431751 IC50 = 790 nM T02703 C35JRN 449021 IC50 = 5000 nM T02703 C40ZOB 544920 IC50 > 50000 nM T02703 CZ3CO7 581866 IC50 > 50000 nM T02703 C8SFX0 708870 IC50 > 50000 nM T02703 C39PAJ 764995 IC50 = 90 nM T02703 CNM06C 1375038 EC50 = 1300 nM T02703 C6U5SR 2733505 IC50 = 5900 nM T02703 C2B8KV 2778315 IC50 = 13200 nM T02703 C70PDZ 2799900 IC50 > 50000 nM T02703 C59BGS 2818222 Ki = 42000 nM T02703 CH5QU8 3016310 IC50 = 14600 nM T02703 C5L7GD 3636377 Ki > 50000 nM T02703 C4VNF7 3792909 IC50 = 86000 nM T02703 C1N8TY 4057533 IC50 = 380 nM T02703 CUI4F5 4247236 IC50 = 80 nM T02703 C97INL 4262401 Ki > 50000 nM T02703 C2OFV8 4452694 IC50 = 4400 nM T02703 C6KW9G 4469991 IC50 = 1700 nM T02703 CS80AZ 6435245 IC50 = 18870 nM T02703 C72QZO 7022594 IC50 > 50000 nM T02703 CLP5G9 8775318 Ki = 4200 nM T02703 CI6O2G 8775930 Ki = 4900 nM T02703 C5GNH3 8776467 Ki = 1400 nM T02703 C5ATV1 9793824 IC50 = 32000 nM T02703 CC52JU 9794039 IC50 = 76 nM T02703 CVZ93W 9795163 IC50 = 6.6 nM T02703 CE62HS 9796600 IC50 = 4600 nM T02703 C4H6JA 9797393 IC50 = 2100 nM T02703 C74XJG 9815372 IC50 = 52000 nM T02703 C3AWZ7 9815642 IC50 = 2360 nM T02703 C96UVG 9815901 Ki = 100000 nM T02703 CN6XG0 9816945 Ki = 3100 nM T02703 CCS6E5 9819003 IC50 = 307400 nM T02703 CR6O0C 9823449 IC50 = 6400 nM T02703 CX7E2G 9823715 IC50 = 3900 nM T02703 CHIO18 9834486 IC50 = 12700 nM T02703 CP21FS 9837291 IC50 = 4500 nM T02703 CBZ95E 9837386 IC50 = 5700 nM T02703 CQF37H 9839201 IC50 = 592 nM T02703 CP2IL5 9842658 Ki = 160 nM T02703 CZMF39 9873870 IC50 = 130000000 nM T02703 CAM64J 9881505 IC50 > 100000 nM T02703 C5DI3E 9896804 IC50 = 10 nM T02703 C0JHT5 9905692 IC50 = 1767 nM T02703 CEF5Q9 9907534 IC50 = 214200 nM T02703 CR49WY 9920741 IC50 = 2700 nM T02703 CAZH53 9920892 IC50 = 34500 nM T02703 C5T7UK 9921294 IC50 = 51 nM T02703 C9MDU2 9921865 IC50 = 600 nM T02703 CBA1D9 9927237 IC50 = 1080 nM T02703 C1LGZ2 9930200 IC50 = 330 nM T02703 C3PH5S 9931834 IC50 = 451800 nM T02703 C72OQJ 9942188 IC50 = 110 nM T02703 CGU01Y 9950094 IC50 = 53 nM T02703 C2I1JH 9950891 IC50 = 27 nM T02703 C29DGM 9951410 IC50 = 78 nM T02703 CY9Q2M 9966187 IC50 = 4 nM T02703 C7ZK5J 9966516 IC50 = 5.4 nM T02703 CJ4RF3 9969613 IC50 = 55 nM T02703 C1YG4Z 9990159 IC50 = 51 nM T02703 CNB2L4 9991061 Ki = 1900 nM T02703 CRD49Q 9991876 IC50 = 33000 nM T02703 CW0Q5C 9999752 IC50 = 590 nM T02703 C0Z2GX 10011896 IC50 = 140 nM T02703 C74TYX 10013642 IC50 = 89 nM T02703 CL3Y5Z 10020993 IC50 = 530 nM T02703 CYZJ64 10034809 IC50 = 133 nM T02703 C7YM4U 10060017 Ki = 600 nM T02703 C04PIY 10068163 IC50 = 250 nM T02703 CS7I1H 10068818 IC50 = 37000 nM T02703 CQB60W 10069033 IC50 = 2200 nM T02703 C38BUK 10077245 IC50 = 101200 nM T02703 C58LCS 10103217 IC50 > 50000 nM T02703 C0DW3A 10103242 IC50 = 420 nM T02703 C3GVU2 10104005 Ki = 90 nM T02703 C3E6CS 10130282 IC50 = 1100 nM T02703 CNU2C3 10133975 IC50 > 10000 nM T02703 C9Z1HS 10149857 IC50 = 38.9 nM T02703 C3N9PS 10154127 IC50 = 40000 nM T02703 C5F8TG 10157080 IC50 = 90 nM T02703 CG43FV 10158280 IC50 > 10000 nM T02703 CM4WK8 10161494 IC50 = 830 nM T02703 CHT12V 10171540 IC50 = 144.54 nM T02703 CD5NH1 10172593 IC50 = 724.44 nM T02703 CJ97GV 10176386 Ki = 480 nM T02703 CFN05B 10180625 IC50 = 450 nM T02703 C7NV2T 10192988 IC50 = 380.19 nM T02703 C4GOJ8 10198117 IC50 = 1100 nM T02703 CHF49M 10215218 IC50 = 512.86 nM T02703 CHVY18 10219750 IC50 = 32000 nM T02703 CK7GN4 10219896 IC50 = 7840 nM T02703 CA68IC 10220131 IC50 = 8750 nM T02703 CZ56SI 10220135 IC50 = 2500 nM T02703 C1FZR9 10220855 IC50 = 1900 nM T02703 C3NPV0 10221335 IC50 = 120 nM T02703 C2LC9R 10222998 IC50 = 92 nM T02703 CAEK83 10248425 IC50 = 580 nM T02703 C8P7WJ 10263292 IC50 = 15000 nM T02703 CBP8Q2 10265375 IC50 = 79000 nM T02703 CVTQ48 10286162 IC50 = 2290.87 nM T02703 C1O4SQ 10292778 IC50 = 74 nM T02703 CN42PW 10308710 IC50 = 186.21 nM T02703 CS8T6Z 10313224 IC50 = 9 nM T02703 C9XQF2 10313251 IC50 = 9800 nM T02703 C0YQK9 10313340 IC50 = 900 nM T02703 CJ3W7S 10330523 IC50 = 12000 nM T02703 C31AYP 10330543 IC50 = 2300 nM T02703 CNKY10 10330544 IC50 = 2100 nM T02703 C7HK2M 10332472 IC50 > 500000 nM T02703 C9P7SQ 10354581 IC50 = 300000 nM T02703 CWDA37 10358114 IC50 = 517 nM T02703 C92DOJ 10390369 IC50 = 0.38 nM T02703 CALW76 10398017 IC50 = 4500 nM T02703 CIHA04 10398629 Ki = 2600 nM T02703 C4P8EC 10400619 IC50 = 14000 nM T02703 CR47JC 10411355 IC50 = 14000 nM T02703 CK7FE5 10445220 IC50 = 350000000 nM T02703 C7E2VQ 10452321 IC50 = 13000 nM T02703 CG94NE 10488346 IC50 = 3200 nM T02703 CB81CA 10489359 IC50 = 14000 nM T02703 C15IWF 10496245 Ki = 2000 nM T02703 CTN4R7 10514976 Ki = 63000 nM T02703 C56DVA 10524594 Ki = 120 nM T02703 C8MIC9 10537022 Ki = 10000 nM T02703 CDY6I3 10538489 Ki = 22000 nM T02703 C8QN6S 10540046 IC50 = 10715.19 nM T02703 C1JMC7 10552176 IC50 = 200 nM T02703 C0JF6I 10575453 IC50 = 400000 nM T02703 C2X0EI 10584290 IC50 = 500 nM T02703 CJG9L3 10607934 Ki = 2500 nM T02703 C2BZ7Q 10608524 Ki = 3200 nM T02703 C1D6GY 10630840 IC50 = 5800 nM T02703 CJD2U9 10630842 IC50 = 3400 nM T02703 CZR04I 10631254 Ki = 23000 nM T02703 C9IVH2 10631255 Ki = 22000 nM T02703 C18YCZ 10632442 Ki = 2400 nM T02703 CNYF76 10634991 Ki = 4700 nM T02703 CZ7QR6 10655660 IC50 > 100000 nM T02703 CCU7H9 10656678 Ki = 25000 nM T02703 C7R3TC 10656792 IC50 = 9200 nM T02703 C9R0NE 10680179 Ki = 2900 nM T02703 COWH50 10688427 Ki > 50000 nM T02703 C94OWI 10702801 IC50 = 190 nM T02703 CF84US 10704325 Ki = 29000 nM T02703 C5CSV1 10727897 Ki = 54000 nM T02703 C3ON1R 10736195 Ki = 17000 nM T02703 C2KEY4 10753994 Ki = 28000 nM T02703 CL38ZM 10755655 Ki = 6600 nM T02703 CGTX82 10761718 Ki = 21 nM T02703 CM2ZI5 10773629 IC50 = 1600 nM T02703 CU5WR9 10788294 Ki = 3400 nM T02703 CGY24Z 10797080 IC50 = 7900 nM T02703 C8YXF1 10797487 Ki = 23000 nM T02703 CHNS51 10797903 Ki = 1900 nM T02703 C5CE9H 10799502 IC50 = 5900 nM T02703 CXZ1W9 10800554 Ki = 3200 nM T02703 CV2ER7 10800919 IC50 = 200 nM T02703 C56AMX 10810281 Ki = 37000 nM T02703 C9F4GI 10822632 IC50 = 8700 nM T02703 CHND09 10823019 Ki = 44000 nM T02703 CMOE80 10825489 Ki = 55000 nM T02703 CJO21R 10845319 IC50 = 5800 nM T02703 CQ7A0W 10882498 IC50 = 106200 nM T02703 CB3CI1 10898715 IC50 = 1000 nM T02703 CM0L3R 10899960 IC50 = 200 nM T02703 CNB4I0 10922301 IC50 = 400 nM T02703 C3IF0R 10925337 IC50 = 47 nM T02703 C93IGZ 10948273 IC50 = 280500 nM T02703 C8LVM1 10977064 IC50 = 300000000 nM T02703 CN7ZJ2 11007884 IC50 = 76 nM T02703 C1WY6T 11010340 IC50 = 2 nM T02703 CX5G2O 11013353 IC50 = 67 nM T02703 CTL03M 11020380 IC50 = 20 nM T02703 C0EK3A 11034111 IC50 = 35 nM T02703 CM36UC 11058021 IC50 = 48 nM T02703 C2MQE0 11075828 IC50 = 1200 nM T02703 C60TVY 11098403 IC50 = 300 nM T02703 C3BVI2 11139807 IC50 = 50 nM T02703 CH6Y1F 11149707 IC50 = 350 nM T02703 CR0JK9 11159816 IC50 = 66 nM T02703 C2X1GP 11161781 IC50 = 89 nM T02703 C2BPQ8 11175135 IC50 = 357.7 nM T02703 C1CH0E 11194833 IC50 = 9.3 nM T02703 COC82L 11194834 IC50 = 34 nM T02703 C46FGL 11210360 IC50 = 2200 nM T02703 COBY89 11229270 IC50 = 21 nM T02703 CAWM24 11240701 IC50 = 22 nM T02703 CQV6W7 11256080 IC50 = 2850 nM T02703 CLN3E1 11267277 IC50 = 450 nM T02703 C6BM4C 11268382 IC50 = 5800 nM T02703 CFN1Y0 11310025 IC50 = 340 nM T02703 C5XS3F 11348978 IC50 = 2367 nM T02703 C6F7WD 11357119 IC50 = 13000 nM T02703 C8WF4O 11369870 IC50 = 3800 nM T02703 CTW93U 11390106 IC50 = 47800 nM T02703 CY03GF 11401263 IC50 = 21 nM T02703 CV97DZ 11426929 IC50 = 530 nM T02703 C9SOQ7 11428573 IC50 = 1280 nM T02703 CIK5B2 11438569 IC50 = 2067 nM T02703 C0YOI9 11473924 IC50 = 9380 nM T02703 C2AW4O 11480938 IC50 = 80 nM T02703 C10SLI 11480939 IC50 = 9.4 nM T02703 CHUP59 11481471 IC50 = 21400 nM T02703 CSBK19 11486109 IC50 = 5750 nM T02703 CP84JR 11495366 EC50 > 100000 nM T02703 C1RU2I 11496223 EC50 = 6 nM T02703 CB43EZ 11502103 EC50 = 29 nM T02703 CP7RX2 11523510 EC50 > 100000 nM T02703 C4JDI3 11524048 EC50 = 2300 nM T02703 CI8B3S 11531856 EC50 = 9 nM T02703 C74RYA 11532340 EC50 = 80 nM T02703 CO8SQ4 11532357 EC50 = 34 nM T02703 C9F6KY 11538267 EC50 = 48 nM T02703 CE1G4D 11539024 EC50 = 4 nM T02703 C2KWX7 11546144 EC50 = 81 nM T02703 CIEU85 11561546 EC50 = 9 nM T02703 CT1Z7W 11575808 EC50 = 4000 nM T02703 CWB4J7 11582528 EC50 = 36 nM T02703 C09EFX 11589024 EC50 = 290 nM T02703 CBR5I2 11590027 EC50 = 59 nM T02703 C46KUP 11596038 EC50 = 293 nM T02703 C2KVY7 11596934 EC50 = 30 nM T02703 C0RTF7 11609610 EC50 > 100000 nM T02703 CDC1M2 11610728 EC50 = 6300 nM T02703 CK04AC 11624646 EC50 = 360 nM T02703 CSI50Y 11625423 EC50 = 12 nM T02703 C9E6TG 11631971 EC50 > 100000 nM T02703 C0MHE1 11633531 EC50 = 14 nM T02703 CWG4J9 11639946 EC50 = 9 nM T02703 CL7Q3I 11646432 EC50 = 8 nM T02703 C4F0CK 11646596 EC50 = 14 nM T02703 CA6D9Z 11654166 EC50 = 56 nM T02703 C8UJ1K 11695590 EC50 > 100000 nM T02703 CM7YA3 11703771 EC50 = 760 nM T02703 CTFW32 11740318 IC50 = 72 nM T02703 C5I6PB 11744927 IC50 = 18000 nM T02703 CD1MV5 11824337 IC50 = 39 nM T02703 CQ5RJ9 11957582 IC50 = 1600 nM T02703 CG63IC 12109769 IC50 = 5900 nM T02703 CS5D0P 12404013 IC50 = 810 nM T02703 CLVQ03 12449028 IC50 > 100000 nM T02703 C2NX4W 12709336 IC50 > 50000 nM T02703 CNJ76X 12778905 IC50 = 26000 nM T02703 C4XK7S 12778908 IC50 = 500 nM T02703 CEJ53H 12778910 IC50 = 2100 nM T02703 CO7T1N 12969094 IC50 = 14500 nM T02703 CJS38P 13154333 Ki = 1400000 nM T02703 CXA84F 13196077 IC50 > 50000 nM T02703 CZ2D9G 13268358 Ki > 50000 nM T02703 C9D4CW 13302397 IC50 = 4100 nM T02703 C9MC3D 13768254 IC50 = 114.82 nM T02703 CI07KP 13768262 IC50 = 48977.88 nM T02703 CZK9A7 15287360 IC50 = 1300 nM T02703 C96DOX 15381020 IC50 = 700 nM T02703 CSJ32F 15453846 IC50 = 5100 nM T02703 C0O5LD 15453847 IC50 = 6000 nM T02703 CXD53V 15825666 IC50 = 2100 nM T02703 CPF1W0 15871186 IC50 = 29000 nM T02703 COV8E5 15887952 IC50 = 2100 nM T02703 C2ZYA6 15951338 IC50 = 36300 nM T02703 CL0SF3 15951408 IC50 = 26500 nM T02703 C1Q8IV 15951410 IC50 = 155000 nM T02703 CZD78C 16114867 IC50 = 1 nM T02703 CN7UX9 16114868 IC50 = 0.5 nM T02703 C4SAV3 16114992 IC50 = 1 nM T02703 C15YED 16114993 IC50 = 0.55 nM T02703 C9F5HZ 16114994 IC50 = 69 nM T02703 CLJ82X 16114995 IC50 = 0.96 nM T02703 CYB3H0 16114996 IC50 = 2.7 nM T02703 C5S2ZL 16114997 IC50 = 0.5 nM T02703 CD95YZ 16115111 IC50 = 1.4 nM T02703 C6K3QJ 16115112 IC50 = 1 nM T02703 CO27LK 16115113 IC50 = 0.28 nM T02703 CS50AC 16115114 IC50 = 0.93 nM T02703 C3A1NY 16115115 IC50 = 1.1 nM T02703 C3LBY0 16115229 IC50 = 52 nM T02703 C1OAI8 16115230 IC50 = 77 nM T02703 C1Q0HJ 16115231 IC50 = 0.8 nM T02703 CA4FB6 16115232 IC50 = 3.7 nM T02703 C53GCA 16115233 IC50 = 1.5 nM T02703 CSC89E 16115341 IC50 = 25 nM T02703 C1FA9K 16115342 IC50 = 3 nM T02703 C9O5KW 16115343 IC50 = 23 nM T02703 CQM69B 16115344 IC50 = 270 nM T02703 CAI72V 16115345 IC50 = 66 nM T02703 C31OYG 16115346 IC50 > 100 nM T02703 CQTR43 16115347 IC50 > 10000 nM T02703 C0UK6B 16115467 IC50 = 63 nM T02703 C3IHD7 16115468 IC50 = 539 nM T02703 CHWL73 16115469 IC50 = 1805 nM T02703 CBM09X 16115471 IC50 = 66 nM T02703 C7XCU0 16115472 IC50 = 3.5 nM T02703 CPHO74 16115473 IC50 = 0.49 nM T02703 CZ9DE8 16115606 IC50 = 4.1 nM T02703 CO9Y1M 16115607 IC50 = 180 nM T02703 CH4VB8 16115608 IC50 = 100 nM T02703 CZQC34 16115609 IC50 = 25 nM T02703 CSD72G 16115610 IC50 = 8.5 nM T02703 C5YH1A 16115611 IC50 = 5.4 nM T02703 C5F0LV 16115743 IC50 = 34 nM T02703 CVEQ13 16115744 IC50 = 0.75 nM T02703 CFU4V2 16115745 IC50 = 0.28 nM T02703 C97IJK 16115746 IC50 = 0.13 nM T02703 C98LIE 16115747 IC50 = 0.29 nM T02703 C4ED1F 16115748 IC50 = 0.52 nM T02703 CS5CU0 16115894 IC50 = 2 nM T02703 C0N9RS 16115896 IC50 = 0.5 nM T02703 C9CX1M 16115897 IC50 = 10 nM T02703 C7MR3Z 16115898 IC50 = 1 nM T02703 C0GV1U 16115899 IC50 = 0.7 nM T02703 CWM82T 16115900 IC50 = 0.48 nM T02703 CI3BV1 16116043 IC50 = 0.87 nM T02703 CJ0N3H 16116044 IC50 = 0.58 nM T02703 CXT25S 16116045 IC50 = 0.67 nM T02703 C7Q1BZ 16116046 IC50 = 0.8 nM T02703 CP71YZ 16116047 IC50 = 1 nM T02703 CFK7V0 16116169 IC50 = 0.24 nM T02703 C4T6NL 16116170 IC50 = 0.5 nM T02703 CD9B3W 16116171 IC50 = 283 nM T02703 CJK86I 16116172 IC50 > 100 nM T02703 C20BHW 16116173 IC50 = 5.7 nM T02703 C7SWH8 16116174 IC50 = 19 nM T02703 CU9LI5 16116293 IC50 > 100 nM T02703 CY5Z1T 16116294 IC50 = 150 nM T02703 CD50GU 16116295 IC50 = 168 nM T02703 CMKW14 16116296 IC50 = 17 nM T02703 C8XH7J 16116297 IC50 = 885 nM T02703 CDU0B4 16116298 IC50 > 100 nM T02703 CMS47F 16116423 IC50 > 100 nM T02703 C1HD2C 16116424 IC50 = 67 nM T02703 CWM1C7 16116425 IC50 = 35 nM T02703 C3Y8KR 16116426 IC50 = 12 nM T02703 CA3L6J 16116427 IC50 = 12 nM T02703 C48ZWL 16116428 IC50 = 1.9 nM T02703 CL1UX6 16116561 IC50 = 300 nM T02703 C0MLO9 16116562 IC50 = 0.12 nM T02703 CQ4Z2O 16116563 IC50 = 0.48 nM T02703 CNMP46 16116564 IC50 = 12 nM T02703 C60FXM 16739321 IC50 = 19 nM T02703 C6Z1DA 16739325 IC50 = 15000 nM T02703 CD3CT0 17793169 IC50 = 3000 nM T02703 C9V0XQ 17897120 IC50 = 360 nM T02703 C3X9JP 17958630 IC50 = 229800 nM T02703 CP2D3I 18356525 Ki = 2500 nM T02703 CKMV50 18428554 IC50 = 2600 nM T02703 CMSA79 18687946 Ki = 10000 nM T02703 C05KOC 18721714 IC50 > 50000 nM T02703 CY28GR 18721729 IC50 > 50000 nM T02703 C9SRI6 18785778 IC50 = 3600 nM T02703 CS76LE 18785786 IC50 = 2700 nM T02703 C4EOC0 18785787 IC50 = 730 nM T02703 CYX62M 18785788 IC50 = 9000 nM T02703 C8XIU6 18785794 IC50 = 2800 nM T02703 CH4QG0 18785802 IC50 = 3500 nM T02703 CG8ZV1 18785805 IC50 = 190 nM T02703 CEMR08 18785810 IC50 = 28000 nM T02703 CHBN50 18785824 IC50 = 150 nM T02703 CCM32F 18785825 IC50 = 2700 nM T02703 C80CGE 18785840 IC50 = 8300 nM T02703 C1JMD3 18785851 IC50 = 5500 nM T02703 CRZ4G5 18785857 IC50 = 880000000 nM T02703 CH26IT 18785878 IC50 = 40 nM T02703 CZ0F5Y 18785885 IC50 = 350000000 nM T02703 CIU32E 18785892 IC50 = 1600 nM T02703 CFLJ71 18785905 IC50 = 4700 nM T02703 C1U9RA 18785910 IC50 = 150 nM T02703 CI8Z7F 18785933 IC50 = 110 nM T02703 CTEZ46 18785938 IC50 = 2700 nM T02703 CY7EO4 18800758 IC50 = 22000 nM T02703 CW0IX3 18983434 IC50 = 38700 nM T02703 CFB10N 20102781 IC50 = 13400 nM T02703 CHME10 20779190 IC50 = 8700 nM T02703 CBT8Q9 21192715 IC50 ~ 50000 nM T02703 CQZ84B 21192814 IC50 = 10 nM T02703 CN5A8J 21834414 IC50 = 4000 nM T02703 CW2VK6 21878467 IC50 = 25000 nM T02703 C8KHU6 21974956 IC50 = 58000 nM T02703 CH70CD 22133392 IC50 = 20000 nM T02703 CIM70E 22260066 IC50 = 120 nM T02703 CM6LX9 22359150 IC50 = 51000 nM T02703 CDO7Q6 22488535 IC50 = 1.1 nM T02703 CZ3X6F 24745386 Ki > 50000 nM T02703 CBNT78 24745536 Ki > 50000 nM T02703 CPH67W 24764596 Ki = 3900 nM T02703 C02RPF 24782142 EC50 = 380 nM T02703 C2UR8E 24782146 EC50 = 8600 nM T02703 C74IOP 24782646 EC50 = 5900 nM T02703 C40NIF 24782649 EC50 = 12000 nM T02703 CD2T4M 24782902 EC50 = 9300 nM T02703 CFG23E 24782903 EC50 = 1800 nM T02703 CM50WK 24785172 EC50 = 4300 nM T02703 C6U0PV 24785174 EC50 = 730 nM T02703 CD7K3S 24785426 EC50 = 1770 nM T02703 CT2UV6 24785697 EC50 = 1360 nM T02703 C3MWU8 24785698 EC50 = 750 nM T02703 CWK68M 24785700 EC50 = 260 nM T02703 C4TC8F 24785702 EC50 = 8900 nM T02703 CO65CH 24785966 EC50 = 48000 nM T02703 CTLA48 24785968 EC50 = 340 nM T02703 C5VBE0 24787679 IC50 = 5000000 nM T02703 C86KAI 24798098 Ki = 3900 nM T02703 CU7F6Y 24801213 Ki = 10500 nM T02703 CI4FH2 24801722 Ki = 16400 nM T02703 C4CDB0 24801723 Ki = 34100 nM T02703 CPQ15V 24894148 IC50 = 31 nM T02703 CYU1V8 24894149 IC50 = 130 nM T02703 CNX5Q3 24894150 IC50 = 1200 nM T02703 C3QK6V 24894151 IC50 = 720 nM T02703 C6J0NK 24894153 IC50 = 40 nM T02703 C7Q3YX 24894154 IC50 = 40 nM T02703 CV7M1Y 24936091 IC50 = 570 nM T02703 C4Z3KW 24941263 IC50 = 40 nM T02703 CRD9A3 25050247 IC50 = 17 nM T02703 C7GYV5 25050248 IC50 = 200 nM T02703 CR3I9Y 25050394 EC50 = 19 nM T02703 C39DOQ 25050395 EC50 = 200 nM T02703 CEZ2M3 25050549 EC50 = 87 nM T02703 CE76PI 25050550 EC50 = 760 nM T02703 CIO41X 25169119 IC50 = 313000 nM T02703 CW0Q3F 25210996 EC50 = 590 nM T02703 C9T1XJ 25211376 EC50 = 180 nM T02703 CD09PR 25211378 EC50 = 270 nM T02703 CD0F1I 25211400 IC50 = 220 nM T02703 C5K3ZC 25211401 IC50 = 77 nM T02703 C9O3QC 25211403 IC50 = 12 nM T02703 CSG69X 25211404 IC50 = 12 nM T02703 CF79GW 25211493 EC50 = 270 nM T02703 CE9DK7 25211494 EC50 = 170 nM T02703 C0DOS1 25211596 EC50 = 210 nM T02703 CT3ID6 25211597 EC50 = 150 nM T02703 C2UQJ6 25211598 EC50 = 88 nM T02703 C43HVC 25211599 EC50 = 280 nM T02703 CDV7E8 25211804 EC50 = 290 nM T02703 CKI86X 25211805 EC50 = 190 nM T02703 CHW2X0 25211910 EC50 = 91 nM T02703 CW0Q7Y 25212125 IC50 = 13 nM T02703 C4EF2A 25212418 IC50 = 10 nM T02703 C7ESB2 25231661 IC50 = 250 nM T02703 CJ92GL 25231666 IC50 = 250 nM T02703 CCO21E 25231830 IC50 = 500 nM T02703 CPHU21 42614330 IC50 = 8900 nM T02703 CNV40T 42618036 EC50 = 1100 nM T02703 CH7AS5 42618037 EC50 = 500 nM T02703 C97FDE 42618038 EC50 = 200 nM T02703 C3MJQ4 42618039 EC50 = 13000 nM T02703 C1YO7H 42618040 EC50 = 11 nM T02703 C0B6JO 42618041 EC50 = 240 nM T02703 C20NYG 42618042 EC50 = 62 nM T02703 C3G6HZ 42618043 EC50 = 56 nM T02703 C3C4FA 42618044 EC50 = 100 nM T02703 C2SK5R 42618045 EC50 = 990 nM T02703 CI9PO8 42618046 EC50 = 53 nM T02703 C1V0KI 42618047 EC50 = 350 nM T02703 CXE5C2 42618048 EC50 = 89 nM T02703 C3S4NL 42618049 EC50 = 49 nM T02703 CN6WQ5 42618050 EC50 = 420 nM T02703 C5F6PW 42618052 EC50 = 16 nM T02703 CMQI75 42618053 EC50 = 770 nM T02703 CN34WV 42618054 EC50 = 160 nM T02703 CY26ND 42618055 EC50 > 100000 nM T02703 C28WPD 42618056 EC50 = 1140 nM T02703 CPYS64 42618057 EC50 = 2000 nM T02703 CUB26P 42618058 EC50 > 100000 nM T02703 C5OM0F 42618059 EC50 > 100000 nM T02703 CH81PY 42618060 EC50 = 1300 nM T02703 CR2TG7 42618061 EC50 > 100000 nM T02703 C4QS7B 42618062 EC50 = 170 nM T02703 CAZ25X 42618063 EC50 = 53 nM T02703 CX5NI3 42618064 EC50 = 300 nM T02703 C54TBN 42618065 EC50 = 500 nM T02703 C0I4MK 42618066 EC50 = 2 nM T02703 CGU3N8 42618068 EC50 = 3 nM T02703 C5UN1C 42618069 EC50 = 3 nM T02703 C8JFX2 42618070 EC50 = 26 nM T02703 CGXT53 42618071 EC50 = 840 nM T02703 C4VK0E 42625538 IC50 > 5000 nM T02703 CTGJ85 42625539 IC50 = 731 nM T02703 CZ35MQ 42625540 IC50 > 5000 nM T02703 CN02OS 42625545 IC50 > 5000 nM T02703 CT1NY0 42625693 IC50 > 5000 nM T02703 C9C5TH 44294245 Ki = 96000 nM T02703 CKT5C3 44294421 Ki = 82000 nM T02703 C5MIG4 44302072 IC50 = 46 nM T02703 CYI6D2 44302109 IC50 = 2700 nM T02703 CE9LX0 44302114 IC50 = 950 nM T02703 CR5C8Z 44302148 IC50 = 3900 nM T02703 C1T7UQ 44302150 IC50 = 1600 nM T02703 C3R1FC 44313302 IC50 = 2800 nM T02703 CHD4J9 44313313 IC50 = 60 nM T02703 CWN2P5 44313352 IC50 = 1400 nM T02703 C2OAM9 44313353 IC50 = 50 nM T02703 C27LBK 44313364 IC50 = 170 nM T02703 CRL32W 44313509 IC50 = 510 nM T02703 C0NUT2 44313550 IC50 = 180 nM T02703 CWR7G1 44313551 IC50 = 310 nM T02703 C2YDZ6 44319656 IC50 = 1700 nM T02703 CQYW59 44319709 IC50 = 8100 nM T02703 CO1Z2F 44319710 IC50 = 5100 nM T02703 C54VXO 44319711 IC50 = 1400 nM T02703 CA81IQ 44319778 IC50 = 2600 nM T02703 CD1QB5 44319779 IC50 = 4100 nM T02703 CR3HT4 44319780 IC50 = 12000 nM T02703 C59RGW 44319825 IC50 = 1100 nM T02703 C76IJF 44319826 IC50 = 1100 nM T02703 CY8K0G 44319828 IC50 = 13000 nM T02703 CQ5A4R 44320031 IC50 = 32000 nM T02703 C0PQ4L 44320069 IC50 = 30000 nM T02703 CL42AK 44320084 IC50 = 89000 nM T02703 CV4XW8 44320115 IC50 = 78000 nM T02703 C80ORG 44322605 IC50 = 9260 nM T02703 CCM47P 44328869 Ki = 2500 nM T02703 CZ2BS4 44328871 Ki = 6100 nM T02703 C7FG5O 44328879 Ki > 50000 nM T02703 C4N5IJ 44328899 Ki = 46000 nM T02703 C34CQV 44328929 Ki > 50000 nM T02703 C0BDZ8 44328932 Ki > 50000 nM T02703 CSG52F 44328934 Ki = 20000 nM T02703 CDF12B 44328946 Ki > 50000 nM T02703 CVO68P 44328955 Ki > 50000 nM T02703 CTAF63 44328957 Ki > 50000 nM T02703 C0W1JK 44328968 Ki > 50000 nM T02703 C7GS5O 44328973 Ki = 6300 nM T02703 C14UCS 44328998 Ki > 50000 nM T02703 CEP9D7 44329003 Ki = 17000 nM T02703 CZQ78B 44329038 Ki = 4000 nM T02703 CG6F2P 44329061 Ki = 46000 nM T02703 C8UEJ6 44329070 Ki = 4600 nM T02703 C39GJB 44329072 Ki > 50000 nM T02703 CPOB75 44329074 Ki > 50000 nM T02703 C3OUZ7 44329119 Ki = 15000 nM T02703 CMW2I5 44329128 Ki > 50000 nM T02703 CNZ5T9 44329167 Ki > 50000 nM T02703 CP4ZU0 44329169 Ki > 50000 nM T02703 CW1VT4 44329187 Ki > 50000 nM T02703 C7PG5J 44329191 Ki > 50000 nM T02703 C1TKS5 44329193 Ki > 50000 nM T02703 C86AGM 44329195 Ki = 10000 nM T02703 C25XJI 44329227 Ki = 2000 nM T02703 CV67AL 44329240 Ki > 50000 nM T02703 CEBZ52 44329255 Ki = 1600 nM T02703 CYX4T3 44329820 IC50 = 7400 nM T02703 C1FHY4 44329948 IC50 = 3500 nM T02703 C5W4FL 44329963 IC50 = 1200 nM T02703 CBQ1O0 44329995 IC50 = 15900 nM T02703 C8F5EQ 44341087 IC50 = 2800 nM T02703 CQ0CU9 44341212 IC50 = 26 nM T02703 CU62NQ 44341315 IC50 = 1800 nM T02703 CWQ18O 44341316 IC50 = 1800 nM T02703 C2YC1E 44347417 IC50 = 810 nM T02703 C86PTS 44347432 IC50 = 660 nM T02703 CQ6DG0 44370661 IC50 > 100000 nM T02703 C0FRX8 44370662 IC50 > 100000 nM T02703 C46TVU 44370689 IC50 = 62000 nM T02703 CYI91R 44370690 IC50 > 100000 nM T02703 C9GZB5 44370704 IC50 > 100000 nM T02703 CKQ20Y 44370705 IC50 = 1400 nM T02703 CS4M3D 44370729 IC50 = 8000 nM T02703 CI7K3E 44370730 IC50 = 5400 nM T02703 C6VS9A 44370736 IC50 = 8000 nM T02703 C12SON 44370747 IC50 = 1200 nM T02703 CF5W2Z 44377082 IC50 = 25000 nM T02703 CW0F6J 44377099 IC50 = 2200 nM T02703 C7K8XO 44377152 IC50 = 1400 nM T02703 C6C2YV 44377153 IC50 = 8100 nM T02703 C2NZ1X 44393481 IC50 > 50000 nM T02703 CDSJ39 44393485 IC50 > 50000 nM T02703 C10WEK 44393495 IC50 > 50000 nM T02703 C85GFC 44396192 IC50 > 50000 nM T02703 C4XL3B 44399796 IC50 = 860 nM T02703 C53KME 44399834 IC50 > 5000 nM T02703 CU98HN 44399945 IC50 = 38 nM T02703 CYW0O2 44400067 IC50 = 974 nM T02703 CC60YN 44402119 IC50 = 3300 nM T02703 CK0OG7 44402176 IC50 = 600 nM T02703 CTV04E 44402250 IC50 = 40 nM T02703 CT96AY 44402285 IC50 = 5600 nM T02703 CU6M4D 44402389 IC50 = 110000 nM T02703 C94GAW 44402453 IC50 > 1000000 nM T02703 CDIR71 44402600 IC50 = 4500 nM T02703 CQTC93 44402628 IC50 = 370000 nM T02703 C65GRQ 44420707 IC50 = 11 nM T02703 CVKR85 44420709 IC50 = 33 nM T02703 C4Q2PY 44427236 IC50 = 130 nM T02703 C9GI4X 44427237 IC50 = 220 nM T02703 C6CS0F 44427238 IC50 = 220 nM T02703 CL5I8G 44430315 IC50 = 580 nM T02703 CM9KR2 44430567 IC50 = 1200 nM T02703 CEH14S 44430628 IC50 = 139000 nM T02703 C0WX4U 44430629 IC50 = 141000 nM T02703 CUO30Z 44430631 IC50 = 48000 nM T02703 C90QJT 44430632 IC50 = 91000 nM T02703 CLZ51V 44430633 IC50 = 14000 nM T02703 CWT98D 44430634 IC50 = 6000 nM T02703 C62UWN 44430635 IC50 = 75000 nM T02703 CI8WV0 44430636 IC50 = 64000 nM T02703 CG13ZP 44430637 IC50 > 100000 nM T02703 C43QST 44430638 IC50 = 9000 nM T02703 C8PTS2 44430640 IC50 > 100000 nM T02703 C58QXR 44430641 IC50 > 100000 nM T02703 CBP09C 44450550 IC50 = 1200 nM T02703 CRF8W4 44455594 IC50 = 470 nM T02703 C2Z5TD 44455595 IC50 = 320 nM T02703 CUK8X2 44455597 IC50 = 1500 nM T02703 C4PE7R 44455626 IC50 = 1200 nM T02703 C1E3AV 44455627 IC50 = 660 nM T02703 C05FUP 44455628 IC50 = 290 nM T02703 CQNA79 44455630 IC50 = 660 nM T02703 C4UZH5 44455631 IC50 = 180 nM T02703 CI9S8P 44455659 IC50 = 6700 nM T02703 CSOK53 44455662 IC50 = 390 nM T02703 C34XKU 44455663 IC50 = 160 nM T02703 C50IWU 44455685 IC50 = 32 nM T02703 CEU63N 44455717 IC50 = 5000 nM T02703 C9E7NX 44455718 IC50 = 300 nM T02703 CH9W2F 44455719 IC50 = 100 nM T02703 CG6I8D 44455720 IC50 = 280 nM T02703 CV8JE9 44455746 IC50 = 3200 nM T02703 CEGL71 44455747 IC50 = 250 nM T02703 C8DQV4 44455748 IC50 = 270 nM T02703 CHAZ31 44455749 IC50 = 3800 nM T02703 CPDZ45 44455769 IC50 = 4500 nM T02703 C02SZW 44455770 IC50 = 670 nM T02703 CQ2VA3 44455771 IC50 = 330 nM T02703 C6CYN7 44455794 IC50 = 420 nM T02703 CVMY02 44455795 IC50 = 3700 nM T02703 CQ9W2U 44455796 IC50 = 5100 nM T02703 CN3D9Q 44455797 IC50 = 700 nM T02703 CSIX74 44455821 IC50 = 3700 nM T02703 C03BYA 44565909 EC50 = 9 nM T02703 C8DUG3 44566070 EC50 = 11 nM T02703 CQ0M1T 46865641 IC50 = 1010 nM T02703 CB1Y8N 49796134 IC50 > 1850000 nM T02703 CN8T5X 49796514 IC50 = 780 nM T02703 CB29CM 49797485 IC50 = 350 nM T02703 CM2D5Z 49836940 EC50 = 3700 nM T02703 CZ51GS 49836941 EC50 = 18000 nM T02703 CM2JB5 49836942 EC50 = 2200 nM T02703 C6ZA7M 49836943 EC50 = 800 nM T02703 C1IHW8 49836944 EC50 = 1600 nM T02703 CM10KE 49837060 EC50 = 600 nM T02703 C3J2SH 49837061 EC50 = 540 nM T02703 CP92KI 49837062 EC50 = 18000 nM T02703 C2ZD0V 49837063 EC50 = 460 nM T02703 C1SB6T 49837065 EC50 = 850 nM T02703 CK38CR 49837066 EC50 = 120 nM T02703 CD8GN9 49837170 EC50 = 220 nM T02703 CZJ85F 49864405 IC50 = 400 nM T02703 CQ8KP7 51003749 IC50 = 4 nM T02703 CUQ53T 52918018 IC50 = 9 nM T02703 CTP6U5 52918019 IC50 = 6 nM T02703 C1MYW7 53233132 IC50 = 120 nM T02703 CZWO31 53387025 IC50 = 25700 nM T02703 C6AYE3 53392451 IC50 = 33200 nM T02703 CYC7G3 54579953 IC50 = 1900 nM T02703 CQ8W0K 54580275 IC50 = 200 nM T02703 CC78LW 54583269 IC50 = 5300 nM T02703 C6TN1Y 54583301 IC50 = 9400 nM T02703 CF5Q0W 54583932 IC50 = 110 nM T02703 C9K2UO 54583934 IC50 = 960 nM T02703 CY4F0W 54584873 IC50 = 71 nM T02703 CCF4H5 54587193 IC50 = 14000 nM T02703 C6QK1A 56593711 IC50 = 2600 nM T02703 CXSQ19 56593712 IC50 = 12300 nM T02703 CY70WM 56593713 IC50 = 9300 nM T02703 C48VIC 56593714 IC50 = 8400 nM T02703 C4U6BD 56593857 IC50 = 18400 nM T02703 CC86JF 56659406 IC50 = 154.88 nM T02703 CSBN93 56659435 IC50 = 70.79 nM T02703 C6P5YB 56666339 IC50 > 100000 nM T02703 CDF86T 56669739 IC50 = 54.95 nM T02703 CRZ08C 56673237 IC50 = 776.25 nM T02703 C8TA3D 56679900 IC50 > 100000 nM T02703 C73MZW 56924689 IC50 = 83000 nM T02703 C83REA 56949933 IC50 > 100000 nM T02703 C2DJ7A 56949934 IC50 > 100000 nM T02703 C3B4DI 56949935 IC50 = 1120 nM T02703 C5DK8C 56950062 IC50 = 6790 nM T02703 C13TGD 56950064 IC50 = 3410 nM T02703 CF2VW1 56950067 IC50 = 8940 nM T02703 CHO6F5 56950186 IC50 = 2390 nM T02703 CHQ5S6 56950187 IC50 = 481000 nM T02703 CRG42P 56950331 IC50 = 522000 nM T02703 C6BZ7V 56951568 IC50 = 5 nM T02703 C0UW5Z 57341142 IC50 > 100000 nM T02703 CS2FH5 57341143 IC50 > 100000 nM T02703 C2AUM9 57341144 IC50 > 100000 nM T02703 CX1FQ0 57341332 IC50 > 100000 nM T02703 CN3Y9D 57341333 IC50 > 100000 nM T02703 C3H1GV 57341334 IC50 = 89400 nM T02703 C0Z3JI 57341335 IC50 = 73000 nM T02703 CDU9W0 57341337 IC50 > 100000 nM T02703 CBO89M 57384807 IC50 = 24000 nM T02703 C2TAS4 57385549 IC50 = 14500 nM T02703 CX2TG9 57385550 IC50 = 54100 nM T02703 CVM67R 57385790 IC50 = 54200 nM T02703 COQ83X 57391112 EC50 = 71 nM T02703 C19RIY 57391700 IC50 = 77 nM T02703 C8Z1PA 57391836 IC50 = 21880 nM T02703 CB1NH9 57392807 EC50 = 20 nM T02703 C6FD9C 57393301 IC50 = 33 nM T02703 C6HO3K 57393302 IC50 = 350 nM T02703 C01NAX 57393303 IC50 = 1300 nM T02703 C7TM3R 57393317 IC50 = 61 nM T02703 C6RKY7 57393439 IC50 = 210 nM T02703 C5QMZ6 57393919 IC50 = 1800 nM T02703 C21UDR 57394528 EC50 = 1800 nM T02703 CVC7Z2 57394614 EC50 = 42 nM T02703 CPQ0S7 57394615 EC50 = 90 nM T02703 C9J6IM 57395031 IC50 = 53 nM T02703 CP4TV8 57395168 IC50 = 31 nM T02703 COKU75 57396367 EC50 = 8900 nM T02703 CV7HI9 57396371 EC50 = 5 nM T02703 CL0P6T 57396785 IC50 = 78 nM T02703 C2QS6D 57396941 IC50 = 13 nM T02703 C4BO9G 57398563 IC50 = 11 nM T02703 CAY3X7 57398682 IC50 = 1500 nM T02703 C6GCN5 57398816 IC50 = 29560 nM T02703 C3GTA7 57398818 IC50 = 41020 nM T02703 CBYG46 57398822 IC50 = 33960 nM T02703 C1DCN7 57401588 EC50 = 230 nM T02703 CQ5HU7 57401590 EC50 > 100000 nM T02703 CA3G1U 57403335 IC50 > 100000 nM T02703 CI2DY9 57403339 EC50 = 163 nM T02703 CD9P4Z 57403764 IC50 = 28 nM T02703 C2ONF1 57403909 IC50 = 130 nM T02703 CYQ70T 57403910 IC50 = 43 nM T02703 CM6C1O 57403911 IC50 = 14 nM T02703 CSWV56 57474449 IC50 = 85000 nM T02703 C0L5HT 62706594 IC50 = 55200 nM T02703 CS9KV1 62706598 IC50 = 15000 nM T02703 CX72ZW 62706764 IC50 = 118000 nM T02703 C2PK8Q 66912454 IC50 = 70000 nM T02703 C37DOA 66912484 IC50 > 100000 nM T02703 CPB9C5 66912809 IC50 = 36000 nM T02703 CF0J3M 67340183 IC50 = 41600 nM T02703 C5HSI6 67492912 IC50 = 40500 nM T02703 C9FMX2 67493358 IC50 = 1500 nM T02703 C3UO2F 70686000 IC50 = 6760 nM T02703 C8XAL1 70686831 IC50 = 43500 nM T02703 CWO02R 70688127 IC50 = 19200 nM T02703 C0M6DH 71484435 IC50 = 17900 nM T02703 CIE6A1 71486265 IC50 = 11400 nM T02703 C2Y1CX 71486266 IC50 = 37300 nM T02703 CO8D6C 71486267 IC50 = 10500 nM T02703 C19AXY 71486268 IC50 = 10100 nM T02703 CK0SO4 71486403 IC50 = 5450 nM T02703 C2C0RP 71486404 IC50 = 21200 nM T02703 CS0X2Q 71486405 IC50 = 39300 nM T02703 C7DH8X 71486406 IC50 = 58200 nM T02703 C9VIN3 71486407 IC50 = 36700 nM T02703 CRZ73J 71486408 IC50 = 94000 nM T02703 CW9V2Q 71718237 IC50 = 5000 nM T02703 CXZ71D 76033629 IC50 > 100000 nM T02703 C26ADC 90662876 IC50 = 49000 nM T02703 C3QU2O 90662877 IC50 = 72000 nM T02703 CYUW16 90664333 IC50 = 11000 nM T02703 CRK93Y 90664334 IC50 = 18000 nM T02703 CAUK54 90664335 IC50 = 4610 nM T02703 CR35FV 90664340 IC50 = 11000 nM T02703 CZ8H2M 90664341 IC50 > 100000 nM T02703 CE5H8T 90664346 IC50 > 100000 nM T02703 CVY3L6 90664347 IC50 = 13500 nM T02703 C5RHW1 90664461 IC50 = 29000 nM T02703 C2G0XJ 90664469 IC50 = 17100 nM T02703 CU7Q9V 90664588 IC50 > 100000 nM T02703 C9TLX0 90664602 IC50 = 14000 nM T02703 CN7P3V 90664608 IC50 = 16900 nM T02703 C8LFX7 90664695 IC50 = 72000 nM T02703 CU29TX 90664696 IC50 = 1200 nM T02703 C7FQ5W 90664698 IC50 = 82000 nM T02703 C8X1LA 90664704 IC50 = 32700 nM T02703 C1PHN4 90664711 IC50 = 60000 nM T02703 C6EGO9 90664714 IC50 = 34000 nM T02703 CS65XI 90664715 IC50 = 15700 nM T02703 CJ61NW 90664716 IC50 = 17000 nM T02703 CVXO58 90664722 IC50 > 100000 nM T02703 CE7H6D 90664727 IC50 = 107900 nM T02703 C9Y2FD 90664833 IC50 = 68000 nM T02703 CE3RV1 90664839 IC50 = 12000 nM T02703 CGK56Q 90664840 IC50 > 100000 nM T02703 C0JM7D 90664841 IC50 = 10000 nM T02703 CL0TG4 90664842 IC50 > 100000 nM T02703 CN3A1P 90664848 IC50 = 58500 nM T02703 C7H8FN 90664849 IC50 > 100000 nM T02703 CA81EW 90664850 IC50 = 1340 nM T02703 C7HGP1 90664855 IC50 > 100000 nM T02703 C8F7HI 90664950 IC50 = 66000 nM T02703 CHA2T6 90664963 IC50 = 9800 nM T02703 CJ01LW 90664969 IC50 = 35000 nM T02703 CF14BZ 90665089 IC50 = 15000 nM T02703 CI4H7Y 90665090 IC50 = 21000 nM T02703 C7PHT4 90665099 IC50 = 58200 nM T02703 C0LM7T 90665100 IC50 > 100000 nM T02703 CY4F6W 90665101 IC50 > 100000 nM T02703 C57NEK 90665196 IC50 = 7600 nM T02703 C3E6MO 90665203 IC50 = 95100 nM T02703 C79CZW 90665204 IC50 = 22000 nM T02703 C2WUY8 90665205 IC50 = 1800 nM T02703 CK62BX 90665207 IC50 > 100000 nM T02703 C02PLA 90665208 IC50 > 100000 nM T02703 CB63ER 90665216 IC50 = 20000 nM T02703 C6RP0B 90667495 IC50 = 60100 nM T02703 CP1L2Q 90667496 IC50 = 57500 nM T02703 CVY5B9 90667497 IC50 = 10000 nM T02703 C4AU9H 90667498 IC50 = 18200 nM T02703 C79IVX 90667499 IC50 = 23000 nM T02703 C8US9C 90667500 IC50 = 100000 nM T02703 CTVK43 90667501 IC50 = 28300 nM T02703 C0QWS6 102068208 IC50 = 2980 nM T02703 C0O9XI 102259962 IC50 = 8450 nM T02703 C7C9DU 127046260 IC50 = 130000 nM T02703 C6HI1S 127047637 IC50 = 710000 nM T02703 CQI26T 127047755 IC50 = 350000 nM T02703 C9QJ2I 127047967 IC50 = 770000 nM T02703 CIO56U 127047968 IC50 > 1000000 nM T02703 CCGY27 127048125 IC50 = 880000 nM T02703 CTL8B5 130449158 Ki = 3501 nM T02703 C76NBO 135409922 IC50 = 10570 nM T02703 C83ZLX 135449023 IC50 = 37440 nM T02703 C7O9XT 135458572 IC50 > 100000 nM T02703 C5H2QR 135674618 IC50 > 500000 nM T02703 C8MN2E 135973134 IC50 > 500000 nM T02703 CMCS36 136035301 IC50 = 122700 nM T02703 CPC52T 136035302 IC50 > 500000 nM T02703 COA8D6 136109078 IC50 > 500000 nM T02703 CHC62Q 136109080 IC50 > 500000 nM T02703 CB4UO8 136109082 IC50 = 374200 nM T02703 CL41DA 137530114 Ki = 1312 nM T02703 C9USH3 137530118 Ki = 2509 nM T02703 CDKB20 137530119 Ki = 3059 nM T02703 CSR3F0 137530120 Ki = 1635 nM T02703 CA39SN 137530121 Ki = 2222 nM T02703 CH1S5L 137530126 Ki = 1780 nM T02703 CF0K6Q 145985455 IC50 = 29230 nM T02703 CN8JM9 146025975 Ki = 21100 nM T02703 CYOA91 146025976 Ki = 43900 nM T02703 CS0BW8 146025977 Ki = 29400 nM T02703 C4S1ZP 146025979 Ki = 24600 nM T02703 C8RWQ4 146025980 Ki = 34800 nM T02703 CCP8X4 155513324 Ki = 3550 nM T02703 CS2UQ8 155535525 IC50 = 7800 nM T02703 C7ZTA4 155540835 Ki = 29900 nM T02703 COAM39 155543079 Ki = 6940 nM T02703 CP59NI 4479245 Ki > 3000000 nM T02703 D00EVC 10197851 IC50 = 28 nM T02703 D00GYE 42625618 IC50 = 170 nM T02703 D00KOE 18983431 IC50 = 3500 nM T02703 D00TDJ 44430622 IC50 = 97000 nM T02703 D01EHS 15552206 IC50 = 3000 nM T02703 D01ILO 15689 IC50 = 900 nM T02703 D01MEA 22617750 IC50 = 500 nM T02703 D01RGM 3311 Ki = 37000 nM T02703 D01TDG 347590 Ki = 870 nM T02703 D01XOR 44396191 IC50 = 1100 nM T02703 D01YNT 10012278 IC50 = 890 nM T02703 D02ELA 107984 Ki = 340 nM T02703 D02EOF 10725313 IC50 = 500 nM T02703 D02KKU 12313704 IC50 = 37000 nM T02703 D02MFQ 10606829 IC50 = 9800 nM T02703 D02TMX 9855524 IC50 = 10 nM T02703 D02TYS 44396204 IC50 = 1200 nM T02703 D02ZGN 42625616 IC50 = 1776 nM T02703 D03CAJ 10375155 IC50 = 152 nM T02703 D03FJM 10198326 IC50 = 7600 nM T02703 D03JXX 10261068 IC50 = 300 nM T02703 D03ODQ 15463448 IC50 = 11800 nM T02703 D03QMU 10104379 IC50 = 500 nM T02703 D03QSQ 19049087 IC50 = 10200 nM T02703 D03WOZ 1893 IC50 = 5800 nM T02703 D04QFO 44393534 IC50 > 50000 nM T02703 D05APC 19049123 IC50 = 300 nM T02703 D05PZA 25231659 IC50 = 200 nM T02703 D05SCE 400010 IC50 = 0.2 nM T02703 D05VAB 9886249 IC50 = 37 nM T02703 D06JZQ 42625621 IC50 = 685 nM T02703 D06VYU 10198539 IC50 = 190 nM T02703 D07BLJ 44322961 IC50 = 13100 nM T02703 D07INO 18428457 IC50 = 1200 nM T02703 D07MFH 44323014 IC50 = 6660 nM T02703 D07OQX 9812839 IC50 = 5200 nM T02703 D07PYV 10439 IC50 = 1900 nM T02703 D07VFC 42625451 IC50 = 220 nM T02703 D08ALG 9793728 IC50 = 2000 nM T02703 D08CMQ 18721725 IC50 = 320 nM T02703 D08FXW 42625617 IC50 = 57.6 nM T02703 D08ISP 19049152 IC50 = 13100 nM T02703 D08JSR 3287412 IC50 = 25000 nM T02703 D08PZX 15463450 IC50 = 1200 nM T02703 D08WEI 18721726 IC50 = 810 nM T02703 D09BKV 15463449 IC50 = 290 nM T02703 D09NRX 18721724 IC50 = 310 nM T02703 D0AO5D 1433 Ki = 140 nM T02703 D0C1OB 12778904 IC50 = 4100 nM T02703 D0D0TO 85237 IC50 = 300 nM T02703 D0D2WC 17892465 IC50 = 23000 nM T02703 D0D3CJ 10308091 IC50 = 81.28 nM T02703 D0D7PK 3268009 IC50 = 16 nM T02703 D0D9LT 12778906 IC50 = 1300 nM T02703 D0DI7W 9793827 IC50 = 200 nM T02703 D0G4ZL 19049163 IC50 = 1200 nM T02703 D0I3ZP 44396203 IC50 = 160 nM T02703 D0I7VD 5139 IC50 = 160 nM T02703 D0IR4Y 9995251 IC50 = 701 nM T02703 D0J2RI 19049061 IC50 = 930 nM T02703 D0J7NS 15887953 IC50 = 200 nM T02703 D0K1CM 10749191 IC50 = 10000 nM T02703 D0K4SV 4102304 IC50 = 14000 nM T02703 D0K4YY 44399940 IC50 = 528 nM T02703 D0L9SL 44322997 IC50 = 2430 nM T02703 D0LB9U 44322572 IC50 = 979 nM T02703 D0LE6N 19049158 IC50 = 3100 nM T02703 D0M4BM 23042899 IC50 = 1800 nM T02703 D0N3HU 15463447 IC50 = 1400 nM T02703 D0N8EU 173566 IC50 = 14000 nM T02703 D0O3XZ 1533 IC50 = 10 nM T02703 D0O9II 189081 IC50 = 2900 nM T02703 D0OW8M 9797857 IC50 = 71 nM T02703 D0R9KX 44399941 IC50 = 186 nM T02703 D0S7MJ 25231669 IC50 = 450 nM T02703 D0SB5H 18721719 IC50 = 3500 nM T02703 D0SJ2Q 10494 IC50 > 40000 nM T02703 D0U8OA 42625452 IC50 = 282 nM T02703 D0U8TM 44622822 IC50 = 400000 nM T02703 D0V9FZ 439202 Ki = 220000 nM T02703 D0VN7G 44393480 IC50 > 50000 nM T02703 D0W9UV 21507 IC50 = 45 nM T02703 D0X2XQ 10467406 IC50 = 46000 nM T02703 D0X5QJ 1649 IC50 = 290 nM T02703 D0X6MB 9942127 IC50 = 1500 nM T02703 D0X6QY 19049121 IC50 = 160 nM T02703 D0XJ1C 10396852 IC50 = 20 nM T02703 D0Y8DZ 10130105 IC50 = 1200 nM T95842 C14OIP 5282539 Ki = 0.08 nM T95842 CAMH93 5282542 Ki = 0.0955 nM T95842 CF2U9Y 5282544 Ki > 199.53 nM T95842 CO16PV 5282545 Ki = 3.311 nM T95842 CD5QS8 5282546 Ki = 5.495 nM T95842 CT6L0C 5282547 Ki = 0.35 nM T95842 C72MTB 5282548 Ki = 3.388 nM T95842 C6C0UY 5282549 Ki = 0.79 nM T95842 CA5YE0 5282550 Ki = 15.49 nM T95842 CAK3G1 5282551 Ki = 0.33 nM T95842 C5KZ9F 9805776 Ki = 0.52 nM T95842 CXS21P 10142377 Ki = 1.7 nM T95842 C6OH0I 10184529 Ki = 0.43 nM T95842 CFUO45 10184774 Ki = 3.2 nM T95842 CJ1O9P 10185917 Ki = 0.09 nM T95842 C3FN5E 10226546 Ki = 1.2 nM T95842 C37LJV 16102853 Ki = 0.81 nM T95842 C01OYF 16102854 Ki = 117 nM T95842 CB35IZ 16102855 Ki > 190 nM T95842 C6XUZ0 16102856 Ki = 29 nM T95842 CEF3A0 16102867 Ki = 59 nM T95842 C91AZO 16102868 Ki = 0.31 nM T95842 CTKI60 24825250 Ki = 6 nM T95842 CG25XE 24825251 Ki = 2.2 nM T95842 CH18NJ 24825252 Ki = 13 nM T95842 CI52AU 24825253 Ki = 3.2 nM T95842 CI1M8P 24825254 Ki = 6 nM T95842 CU86CM 24825255 Ki = 2.7 nM T95842 CRZ1K5 24825256 Ki = 0.29 nM T95842 C5Q3ZJ 24825257 Ki = 0.42 nM T95842 CL86QS 24825258 Ki = 0.68 nM T95842 CM92PE 24825259 Ki = 6.5 nM T95842 CV1P6N 24825260 Ki = 12 nM T95842 CUX47I 24825261 Ki = 1.1 nM T95842 C7G6OT 24825262 Ki = 1.9 nM T95842 CJ14IQ 24825263 Ki = 9.2 nM T95842 CO0SF1 24825264 Ki = 8.7 nM T95842 CV16QE 24825265 Ki = 37 nM T95842 CCHL59 24825266 Ki = 3.5 nM T95842 C1B8TF 24825267 Ki = 5.3 nM T95842 C06COB 24825268 Ki = 3.9 nM T95842 C47QTG 24825269 Ki = 4.7 nM T95842 CJ16YD 24825270 Ki = 6.6 nM T95842 CO1BL7 24825271 Ki = 16 nM T95842 CV0UB1 24825272 Ki = 26 nM T95842 CIB8U9 122212031 EC50 = 1000 nM T95842 C78CVX 122212032 EC50 = 690 nM T95842 CZ30WH 122212034 EC50 = 55 nM T95842 CRZL02 122212035 EC50 = 60 nM T95842 CBHS96 127048413 EC50 = 0.16 nM T95842 C8Q9PL 127048414 EC50 = 100 nM T95842 C3NHY6 127048415 EC50 = 0.8 nM T95842 C2D9TA 127049085 EC50 = 11 nM T95842 C7N2BY 127049401 EC50 = 4 nM T95842 CSAF25 127052514 EC50 = 500 nM T95842 CN8MJ1 127052807 EC50 = 0.8 nM T95842 CCV59R 127052808 EC50 = 420 nM T95842 C0ZWJ8 127052809 EC50 = 24 nM T95842 CCS7U2 127052810 EC50 = 520 nM T95842 CWJ7O5 127053099 EC50 = 0.8 nM T95842 CI47OQ 5282543 Ki = 23 nM T91761 D09KTS 24821094 IC50 = 3 nM T91761 D0E6XR 3062316 IC50 = 228 nM T91761 D02NNV 3038525 IC50 > 10000 nM T91761 D02TUL 118115473 Ki = 26.9 nM T91761 D08AOZ 86582336 IC50 = 410 nM T91761 D0E3TC 44259 IC50 = 10 nM T91761 D0G5XV 135565884 IC50 = 56 nM T91761 D0LF1U 5287969 IC50 > 14850 nM T91761 D0S5RC 3025986 IC50 > 40000 nM T91761 D0YB3W 156414 IC50 = 5650 nM T91761 D03BNU 59604787 IC50 > 10000 nM T91761 D0LF0O 135441202 IC50 = 370 nM T91761 C9VW8M 449054 IC50 > 16000 nM T91761 CED2F1 668334 Ki = 460 nM T91761 CB6R5K 3722581 Ki = 15 nM T91761 CTID76 5282335 IC50 = 29000 nM T91761 CUCE63 5329663 IC50 > 10000 nM T91761 C8SU6K 9806812 IC50 = 1000 nM T91761 CM5Z8X 9869943 IC50 > 10000 nM T91761 CERH18 9871955 IC50 = 540 nM T91761 CV02OT 9914277 IC50 = 970 nM T91761 CQ2S4D 9964914 Ki = 3000 nM T91761 C7YD1X 10048045 IC50 > 25000 nM T91761 CXG4Q9 10110453 IC50 = 4800 nM T91761 CF34HN 10114123 IC50 = 950 nM T91761 CVM07F 10120124 IC50 = 230 nM T91761 C7R9GF 10151801 IC50 = 250 nM T91761 C28JIN 10151831 IC50 = 160 nM T91761 C1Q9PD 10152000 IC50 = 1100 nM T91761 CZ4JE8 10160476 IC50 = 92 nM T91761 CG1FZ5 10162990 IC50 = 270 nM T91761 C6QU7V 10163233 IC50 = 1300 nM T91761 C2G5HY 10165201 IC50 = 260 nM T91761 C9J2KW 10181704 IC50 = 690 nM T91761 CK0SX4 10194689 IC50 = 1600 nM T91761 C5PKO2 10195094 IC50 = 370 nM T91761 CD18OB 10195108 IC50 = 69 nM T91761 CXI97Z 10195393 IC50 = 7400 nM T91761 CF84LX 10195646 IC50 = 60 nM T91761 CGM5W0 10217158 IC50 = 390 nM T91761 CKH5C7 10217329 IC50 = 7200 nM T91761 C9R7FB 10224336 IC50 = 190 nM T91761 C2ODX6 10228329 IC50 = 76 nM T91761 CQ3Z6X 10230606 IC50 = 81 nM T91761 CSGD16 10246246 IC50 > 7000 nM T91761 C89JTD 10288201 IC50 = 330 nM T91761 CXS48F 10288395 IC50 = 110 nM T91761 C4QR0P 10301758 IC50 = 940 nM T91761 C47LSO 10310783 IC50 = 140 nM T91761 C5TYO0 10310880 IC50 = 730 nM T91761 CJ7U4I 11161778 IC50 = 17000 nM T91761 C2W5RC 11235063 IC50 > 50000 nM T91761 CRK56F 11237786 IC50 = 650 nM T91761 CBOP58 11293798 Ki > 10000 nM T91761 CJ8A6Y 11341428 IC50 = 820 nM T91761 C26BZX 11362471 Ki > 10000 nM T91761 CWXB93 11397177 Ki > 10000 nM T91761 CEP8N2 11489351 IC50 = 2 nM T91761 CRU9D3 11508262 Ki = 210 nM T91761 C4BK1O 11514905 Ki > 30000 nM T91761 CKX45I 11536964 Ki > 6000 nM T91761 CTG83F 11539329 Ki > 3800 nM T91761 CPW27V 11581044 Ki = 120 nM T91761 CMIL86 11590363 Ki > 3800 nM T91761 CJU5W6 11611103 Ki = 112 nM T91761 CI8CR3 11623444 Ki = 1300 nM T91761 C3UDF2 11623669 Ki = 1200 nM T91761 CK34LS 11632737 IC50 > 50000 nM T91761 C9T6SC 11640926 Ki > 3800 nM T91761 C5B6KR 11660004 Ki = 280 nM T91761 CLXI20 11675164 Ki = 220 nM T91761 CHSL63 11688314 Ki = 530 nM T91761 CU0E8O 11690457 Ki > 10000 nM T91761 CB16DG 11695198 Ki = 2100 nM T91761 CB0AP2 11705863 Ki > 10000 nM T91761 CE49IU 11718919 Ki > 2000 nM T91761 C45EWD 11723489 IC50 > 7000 nM T91761 CFPW41 16007116 Ki > 1500 nM T91761 CKR57M 16086104 IC50 > 5000 nM T91761 C16NRY 16086114 IC50 > 25000 nM T91761 CQG45C 16109001 IC50 = 25000 nM T91761 C1U8XW 16109036 IC50 > 5000 nM T91761 CGC34R 16118737 IC50 > 25000 nM T91761 C0H8UN 16730109 IC50 > 50000 nM T91761 CEW2T0 17501441 Ki > 4 nM T91761 CAF64K 20635205 IC50 = 30 nM T91761 CNLC10 20635235 IC50 = 7 nM T91761 C4PXQ6 20635236 IC50 = 6 nM T91761 C5LS4A 20635249 IC50 = 7 nM T91761 CD04JU 20635261 IC50 = 83 nM T91761 CPQ1F9 20635262 IC50 = 34 nM T91761 C3OH6S 20635263 IC50 = 15 nM T91761 C4XGT7 20635267 IC50 = 370 nM T91761 CTA9W2 20635268 IC50 = 320 nM T91761 CZ4W7A 20635392 IC50 = 2400 nM T91761 C16JNA 20635396 IC50 = 96 nM T91761 C3F4MT 20635404 IC50 = 40 nM T91761 C7NZ2P 20635405 IC50 = 35 nM T91761 C1ITS2 20635410 IC50 = 350 nM T91761 C75ATW 20635412 IC50 = 34 nM T91761 C4DAM0 20635501 IC50 = 250 nM T91761 C1V2MY 20635507 IC50 = 7 nM T91761 CB9E7N 20635510 IC50 = 19 nM T91761 C0XIQ2 20635514 IC50 = 12 nM T91761 COV49P 20635515 IC50 = 14 nM T91761 C2V5RM 20635525 IC50 = 18 nM T91761 CA12GX 20635526 IC50 = 29 nM T91761 CDTH82 20635527 IC50 = 47 nM T91761 CK2X6E 20635530 IC50 = 20 nM T91761 C8T7OA 20635534 IC50 = 9 nM T91761 CM83LK 20635537 IC50 = 260 nM T91761 CA61QF 21083895 IC50 = 9100 nM T91761 C6SL2R 22170396 IC50 = 60 nM T91761 C2FHR8 22170398 IC50 = 90 nM T91761 C0A8BN 22170403 IC50 = 290 nM T91761 CMNU25 22170411 IC50 = 930 nM T91761 CL9IA2 22170419 IC50 = 30 nM T91761 CRK8D4 22170436 IC50 = 210 nM T91761 CH5T9P 22170437 IC50 = 2190 nM T91761 C6JV7W 23400934 IC50 > 7000 nM T91761 CD5S7O 23401001 IC50 > 7000 nM T91761 CF67IQ 23628269 IC50 = 40 nM T91761 C7YG1N 24759534 IC50 = 26 nM T91761 CQNP54 24764449 IC50 = 62 nM T91761 C2UOE0 24766030 IC50 > 20000 nM T91761 CY8X0J 24811794 Ki > 10000 nM T91761 C9F1AO 24821023 IC50 = 11 nM T91761 CS3Q8B 24995659 IC50 > 2000 nM T91761 C0B7RT 25057409 IC50 > 10000 nM T91761 C0K9HA 25110600 IC50 = 46 nM T91761 CSNC57 25110758 IC50 = 3 nM T91761 C0GOX5 25110759 IC50 = 6 nM T91761 CC2R7S 25110760 IC50 = 7 nM T91761 CL82CU 25110796 IC50 = 4 nM T91761 CHT0B4 25169252 IC50 = 280 nM T91761 CJL25F 25169253 IC50 = 410 nM T91761 C2RX6E 25190503 IC50 = 3 nM T91761 CFN61D 25190504 IC50 = 170 nM T91761 C8LQS3 25190505 IC50 = 26 nM T91761 C20WQJ 25190506 IC50 > 5000 nM T91761 CM61RX 25190507 IC50 = 90 nM T91761 C5UCN3 25190508 IC50 = 2500 nM T91761 CTVK31 25190509 IC50 = 95 nM T91761 CY43QX 25190510 IC50 = 14 nM T91761 C09SGT 25190511 IC50 = 57 nM T91761 C9O0AL 25190512 IC50 = 340 nM T91761 C6RC2N 25190513 IC50 = 130 nM T91761 CA9U5F 25190514 IC50 = 450 nM T91761 C1ZCK4 25190515 IC50 = 170 nM T91761 CBX7Z3 25190516 IC50 = 180 nM T91761 CY3X8L 25190517 IC50 = 10 nM T91761 CONP02 25190518 IC50 = 14 nM T91761 CL81KR 25190519 IC50 = 100 nM T91761 C2I6JX 25190520 IC50 = 15 nM T91761 C8TK1S 25190521 IC50 = 2 nM T91761 CHD51B 25190522 IC50 = 14 nM T91761 C0G9EX 25190523 IC50 = 570 nM T91761 CUJS83 25190524 IC50 = 55 nM T91761 CE3W4R 25190525 IC50 = 140 nM T91761 CIAB51 25190526 IC50 = 1200 nM T91761 CA4Z2Y 25190527 IC50 = 5 nM T91761 C8OW9I 25190528 IC50 = 100 nM T91761 C5PH6D 25190529 IC50 = 740 nM T91761 CZ46JX 25190530 IC50 = 50 nM T91761 CE3T5U 25190531 IC50 = 6 nM T91761 CEHP95 25190532 IC50 = 190 nM T91761 C06LXS 25190533 IC50 = 10 nM T91761 C9RXL3 25190534 IC50 = 2 nM T91761 CC1E3O 25190535 IC50 = 13 nM T91761 C1NZ4D 25190536 IC50 = 81 nM T91761 CNR75T 25190537 IC50 = 380 nM T91761 C7LMI1 25190538 IC50 = 150 nM T91761 CLU7D2 25190539 IC50 = 74 nM T91761 CD2Z1T 25190540 IC50 = 8 nM T91761 CUP7E4 25190541 IC50 = 60 nM T91761 C57KGJ 25190542 IC50 = 10 nM T91761 CF9C5J 25190543 IC50 = 5 nM T91761 C3KJ6P 25190544 IC50 = 2 nM T91761 CU6VA8 25190545 IC50 = 7 nM T91761 CR0JP6 25190546 IC50 = 390 nM T91761 CJLB59 25190547 IC50 = 10 nM T91761 C27RCT 25190548 IC50 = 11 nM T91761 CM7A8T 25190549 IC50 = 6 nM T91761 C3YA7U 25190550 IC50 = 5 nM T91761 C6SE7Y 25190551 IC50 = 65 nM T91761 CPK7E0 25190552 IC50 = 67 nM T91761 CA2K4Q 25190553 IC50 = 13 nM T91761 CWRO62 25190554 IC50 = 58 nM T91761 C5UFS2 25190555 IC50 = 270 nM T91761 C6J2UZ 25190556 IC50 = 30 nM T91761 CMP9A2 25190557 IC50 = 130 nM T91761 CKP50F 25190558 IC50 = 6 nM T91761 CE3W9P 25190559 IC50 = 9 nM T91761 CNBO46 25190560 IC50 = 6 nM T91761 CCP4K9 25190561 IC50 = 42 nM T91761 CYK5Z2 25190562 IC50 = 740 nM T91761 C25JMO 25190563 IC50 = 8 nM T91761 CJ4W6E 25190564 IC50 = 12 nM T91761 CBV3D6 25190565 IC50 = 7 nM T91761 CE9UI6 25190566 IC50 = 37 nM T91761 CAK4E6 25190567 IC50 = 63 nM T91761 CTR6A2 25190568 IC50 = 39 nM T91761 CC40BJ 25190569 IC50 = 75 nM T91761 C7B6OS 25190570 IC50 = 39 nM T91761 CCJY98 25190571 IC50 = 59 nM T91761 C57PDK 25191024 IC50 = 510 nM T91761 CN5E0F 25263283 IC50 = 19000 nM T91761 CB8YN2 44201333 IC50 = 1 nM T91761 C8KNA3 44219632 Ki > 4000 nM T91761 C0VIX4 44219633 Ki > 4000 nM T91761 C39MDP 44410415 IC50 = 5000 nM T91761 CAMH81 44410416 IC50 = 14000 nM T91761 CW4U8D 44410417 IC50 = 4600 nM T91761 CEWY72 44410418 IC50 = 1700 nM T91761 CBZ9G1 44410419 IC50 = 730 nM T91761 CB16MX 44410420 IC50 = 2200 nM T91761 CM4J5W 44410421 IC50 = 2100 nM T91761 C5VR2O 44410424 IC50 = 2420 nM T91761 C32GPA 44410428 IC50 = 1090 nM T91761 C9E7KL 44410430 IC50 = 1030 nM T91761 CL7W3J 44410455 IC50 = 2600 nM T91761 CQLO41 44410456 IC50 = 900 nM T91761 CW7A2I 44410457 IC50 = 39000 nM T91761 C3HK5U 44410461 IC50 = 14800 nM T91761 C1Z3YU 44410513 IC50 > 50000 nM T91761 CQX90C 44410514 IC50 = 1600 nM T91761 CTFW82 44410519 IC50 = 1600 nM T91761 CN2A5F 44410567 IC50 = 600 nM T91761 C9M2AF 44410577 IC50 = 37000 nM T91761 C6SN3R 44410609 IC50 = 380 nM T91761 CKBT38 44410612 IC50 > 50000 nM T91761 C1FMC7 44410613 IC50 > 50000 nM T91761 C8QW6B 44410614 IC50 > 50000 nM T91761 CT6PH4 44410617 IC50 > 50000 nM T91761 CW93VP 44410622 IC50 = 13000 nM T91761 CFQ6I2 44410627 IC50 = 1440 nM T91761 CDB3X8 44410652 IC50 = 260 nM T91761 C6ZMA0 44410656 IC50 = 15000 nM T91761 C1FR5B 44410659 IC50 > 50000 nM T91761 CGA70U 44410660 IC50 > 50000 nM T91761 CB32UG 44410662 IC50 > 50000 nM T91761 C6E0TJ 44410667 IC50 > 50000 nM T91761 CR9LC6 44410668 IC50 = 11200 nM T91761 CARJ28 44410676 IC50 = 5700 nM T91761 CT9G0X 44410737 IC50 = 350 nM T91761 CLVC63 44410741 IC50 = 720 nM T91761 CA7ZC5 44410746 IC50 = 2000 nM T91761 CKI8M1 44412537 IC50 = 600 nM T91761 C8LDU0 44412550 IC50 = 820 nM T91761 C1Y7OA 44412551 IC50 = 3900 nM T91761 CTM8Z6 44412588 IC50 = 22340 nM T91761 CRG1L6 44412606 IC50 > 25000 nM T91761 C4NUK8 44412771 IC50 = 1130 nM T91761 CC0WJ8 44412792 IC50 = 19240 nM T91761 C5G4SU 44413075 IC50 > 50000 nM T91761 CADR04 44413087 IC50 = 46300 nM T91761 CG8NE2 44413088 IC50 = 6060 nM T91761 C7OF0Q 44413100 IC50 = 7070 nM T91761 COH5J0 44413186 IC50 = 34200 nM T91761 CMVT21 44432424 IC50 = 2700 nM T91761 CPX6K4 44432425 IC50 = 62 nM T91761 C6A3NK 44432426 IC50 > 20000 nM T91761 CD4Q5O 44432427 IC50 > 20000 nM T91761 CI95MW 44432428 IC50 > 20000 nM T91761 CJ1FH3 44432429 IC50 = 11000 nM T91761 CW5J2A 44432432 IC50 = 20000 nM T91761 CU90YD 44432433 IC50 = 12000 nM T91761 CA38PO 44432438 IC50 = 11000 nM T91761 CH4DL7 44432439 IC50 > 20000 nM T91761 C46ZFU 44432440 IC50 = 1700 nM T91761 CA98KR 44432441 IC50 = 110 nM T91761 C3VRO9 44557921 IC50 > 10000 nM T91761 CJAV21 44573146 IC50 = 3 nM T91761 CP9E4J 44573266 IC50 = 100 nM T91761 CLA24D 44573267 IC50 = 11 nM T91761 C51CDF 44573268 IC50 = 8 nM T91761 CDT4K9 44573269 IC50 = 940 nM T91761 CD8Q5P 44573306 IC50 = 780 nM T91761 C5CA0V 44573307 IC50 = 2 nM T91761 CNMO98 44573308 IC50 = 2 nM T91761 CAZ59C 44573309 IC50 = 20 nM T91761 C7T3HJ 44573374 IC50 = 4 nM T91761 CPMG47 44573375 IC50 = 2 nM T91761 CT1R3Z 44573376 IC50 = 3 nM T91761 CF3N7G 44573377 IC50 = 140 nM T91761 C6BRV7 44573424 IC50 = 1 nM T91761 CXU7T6 44573425 IC50 = 2 nM T91761 C81CVB 44573426 IC50 = 1 nM T91761 CS27CU 44573427 IC50 = 3 nM T91761 CAYJ73 44573467 IC50 = 1 nM T91761 CN6G1U 44573468 IC50 = 8 nM T91761 CO4N5B 44573469 IC50 = 2 nM T91761 CDU34Y 44573502 IC50 = 3 nM T91761 CY81WI 44573503 IC50 = 660 nM T91761 CM9E7S 44573504 IC50 = 2 nM T91761 C42NEB 44573505 IC50 = 1 nM T91761 CK24OS 44573546 IC50 = 2 nM T91761 C53MYT 44588579 IC50 = 10 nM T91761 CSY05L 44588580 IC50 = 27 nM T91761 CSV19C 44588581 IC50 = 18 nM T91761 CKN87Z 44588582 IC50 = 46 nM T91761 CJB84Y 44588583 IC50 = 8 nM T91761 CI30GZ 44588584 IC50 = 76 nM T91761 C2C6XI 44588606 IC50 = 54 nM T91761 CU4A2I 44588607 IC50 = 3 nM T91761 C6Z3CL 44588719 IC50 = 10 nM T91761 CXN8P2 44588738 IC50 = 5 nM T91761 CNPI73 44588739 IC50 = 10 nM T91761 CK34PA 44588740 IC50 = 25 nM T91761 CL67AQ 44588741 IC50 = 16 nM T91761 C6JVC8 44588765 IC50 = 9 nM T91761 C0C9UI 44588766 IC50 = 3 nM T91761 CT6VG5 44588767 IC50 = 10 nM T91761 CZ1P6B 44588791 IC50 = 12 nM T91761 CWJ92G 44588792 IC50 = 3300 nM T91761 C4U8BY 44588793 IC50 = 56 nM T91761 CU6O3G 44588794 IC50 = 35 nM T91761 C30HRN 44588845 IC50 = 4 nM T91761 CY5T8I 44588846 IC50 = 68 nM T91761 C1YI7Z 44588847 IC50 = 250 nM T91761 CK79TL 44588878 IC50 = 4500 nM T91761 CML1U9 44588879 IC50 = 520 nM T91761 C10BIC 44588880 IC50 > 10000 nM T91761 C3JS6Q 44588881 IC50 = 270 nM T91761 C2VDN8 44588915 IC50 = 16 nM T91761 CSC84A 44588916 IC50 = 4500 nM T91761 C4FIC7 44588917 IC50 = 35 nM T91761 C4Z1DQ 44588918 IC50 = 6 nM T91761 CKB0C7 44588945 IC50 = 89 nM T91761 CG6RP1 44588946 IC50 = 690 nM T91761 CJ6BN1 44588947 IC50 = 2000 nM T91761 CLO50G 44588965 IC50 = 2 nM T91761 CLA8G9 44588966 IC50 = 12 nM T91761 CV03WM 44588967 IC50 = 16 nM T91761 C5I7DE 44588968 IC50 = 73 nM T91761 C82SKN 44588969 IC50 = 9 nM T91761 CTL5U3 44588970 IC50 = 14 nM T91761 CFYP17 44588994 IC50 = 10 nM T91761 CRU7I3 44588995 IC50 = 1100 nM T91761 CQR2N6 44588996 IC50 = 35 nM T91761 C3J7WS 44588997 IC50 = 4 nM T91761 C0UFA7 44588998 IC50 = 61 nM T91761 C4S3ZD 44588999 IC50 = 5 nM T91761 CUY54I 44589015 IC50 = 27 nM T91761 C5RG0W 44589016 IC50 = 1900 nM T91761 C6QFD0 44589017 IC50 = 5 nM T91761 CW2DV3 44589018 IC50 = 18 nM T91761 CEGF45 44589019 IC50 > 20000 nM T91761 CWO6V3 44589020 IC50 > 20000 nM T91761 C6FJ7Y 44589021 IC50 = 7 nM T91761 CXE42M 44589045 IC50 = 23 nM T91761 CC4DW7 44589046 IC50 = 150 nM T91761 CCJM31 44589047 IC50 = 59 nM T91761 C7NRT2 44589048 IC50 = 320 nM T91761 CATZ92 44589049 IC50 = 220 nM T91761 CG1X2R 44589639 IC50 = 170 nM T91761 C7Y2UR 44589640 IC50 = 45 nM T91761 CKU74A 44589641 IC50 = 48 nM T91761 CB06FP 44589642 IC50 = 34 nM T91761 CH4OB9 44589677 IC50 = 81 nM T91761 CU3MJ6 44589678 IC50 = 69 nM T91761 CYDZ59 44589679 IC50 > 10000 nM T91761 CDJ51R 44589680 IC50 = 46 nM T91761 CNI87X 44589716 IC50 = 20 nM T91761 CEZ4C6 44589717 IC50 = 1200 nM T91761 CJ8P0D 44589718 IC50 = 47 nM T91761 CKE0R1 44589719 IC50 = 36 nM T91761 CT3W7G 44589754 IC50 = 6 nM T91761 C7PMB4 44589755 IC50 = 41 nM T91761 CLI17Q 44589756 IC50 = 30 nM T91761 C9MDA8 44589757 IC50 = 27 nM T91761 CK2L6P 44589793 IC50 = 46 nM T91761 CY7HW6 44589794 IC50 = 53 nM T91761 CBW27Y 44589795 IC50 = 3 nM T91761 CO21BJ 44589832 IC50 = 110 nM T91761 CZL1U2 44593710 IC50 = 8 nM T91761 C9B7LK 44593713 IC50 = 4 nM T91761 CY3HW5 46224684 IC50 > 10000 nM T91761 C7H4YM 46865419 IC50 > 10000 nM T91761 CLS29B 46872626 IC50 > 10000 nM T91761 C2O8RZ 46886323 IC50 > 1000 nM T91761 C28ELR 46912278 Ki = 1.585 nM T91761 CD4L7V 46912279 Ki = 0.2512 nM T91761 C7S2HO 46913757 Ki = 0.1995 nM T91761 CT46HI 46913758 Ki = 0.2512 nM T91761 C9L3XR 49838879 IC50 > 50000 nM T91761 C5V9BE 52936431 Ki = 140 nM T91761 CR3X8W 52936432 Ki > 30000 nM T91761 C13LER 52936433 Ki = 170 nM T91761 C1VML8 52936434 Ki = 93 nM T91761 CU1T5C 52936530 Ki = 7 nM T91761 CK69ML 52936531 Ki = 16 nM T91761 CCT6B9 52936532 Ki = 46 nM T91761 CC7SE4 52936533 Ki = 145 nM T91761 CA93FM 52936534 Ki = 11 nM T91761 C9KO7D 52936535 Ki = 23 nM T91761 CEQN27 52936621 Ki = 7 nM T91761 C2A6MX 52936622 Ki = 20 nM T91761 CBH0K9 52936623 Ki = 20 nM T91761 CKF2D5 52936624 Ki = 27 nM T91761 CD4H3S 53354074 Ki > 1000 nM T91761 C8ZRE3 53356518 IC50 = 52 nM T91761 CN9QD7 56643097 IC50 > 10000 nM T91761 CJBL48 56925034 IC50 = 39 nM T91761 C7RDQ8 56925241 IC50 = 5 nM T91761 CT3EW2 59292007 IC50 > 1000 nM T91761 CZ3TG1 59375154 IC50 = 55 nM T91761 CXJ63M 59603829 IC50 = 94 nM T91761 CQEU96 59603842 IC50 = 26 nM T91761 CV63UL 67240318 IC50 > 10000 nM T91761 C5DGR9 69036886 IC50 = 10000 nM T91761 C3GTU1 69762142 IC50 > 10000 nM T91761 C7VJ6A 70647728 IC50 = 96 nM T91761 C5HB9I 71259491 Ki = 0.1 nM T91761 C6D0JX 71259500 Ki = 1.4 nM T91761 CP5O3N 71259506 Ki = 59 nM T91761 C64KQW 71259516 Ki = 6.6 nM T91761 CS92ID 71259555 Ki = 0.93 nM T91761 C2WL5D 71259557 Ki = 44 nM T91761 C7BNF0 71259563 Ki = 27 nM T91761 C4SJ1M 71259597 Ki = 7.8 nM T91761 CC96VO 71259598 Ki = 0.56 nM T91761 CK9MW3 71259641 Ki = 1 nM T91761 C4SPA0 71259651 Ki = 35 nM T91761 CJ4BK2 71259773 Ki = 10 nM T91761 CKH6Z3 71259783 Ki = 580 nM T91761 C1IZT4 71259797 Ki = 36 nM T91761 C9AF8W 71267243 Ki = 0.8 nM T91761 CE5SB7 71267246 Ki = 381 nM T91761 CG7U6V 71267305 Ki = 11 nM T91761 CI0R3A 71267318 Ki = 0.8 nM T91761 C5X2UZ 71267326 Ki = 0.23 nM T91761 C76CXB 71450143 IC50 = 2450 nM T91761 CY8X9L 71450144 IC50 > 100000 nM T91761 C4MBT3 71450145 IC50 = 720 nM T91761 C5YX9S 71450146 IC50 = 2 nM T91761 CYP5D9 71450147 IC50 = 6470 nM T91761 C2PV9H 71450148 IC50 = 1750 nM T91761 C9ID7H 71450149 IC50 = 780 nM T91761 CDLK74 71450150 IC50 = 65000 nM T91761 CA03KS 71450151 IC50 = 21417 nM T91761 CBMZ60 71450184 IC50 = 7457 nM T91761 CCYE35 71450185 IC50 = 4425 nM T91761 C34TYA 71450186 IC50 = 2495 nM T91761 C34MPQ 71451977 IC50 > 100000 nM T91761 CUK4C0 71451978 IC50 = 53650 nM T91761 C1CH6E 71451979 IC50 = 190 nM T91761 CWF2H0 71451980 IC50 = 180 nM T91761 CZL5M2 71451981 IC50 = 210 nM T91761 C0G3FM 71451982 IC50 > 100000 nM T91761 CQR24F 71453784 IC50 = 100 nM T91761 C8BLW0 71453785 IC50 = 10 nM T91761 CPA8Q9 71453786 IC50 = 520 nM T91761 CHM1S9 71453787 IC50 = 1520 nM T91761 CY0C7F 71453788 IC50 = 10880 nM T91761 C94XDU 71453789 IC50 = 36220 nM T91761 CNFQ61 71453790 IC50 > 100000 nM T91761 C3MYB5 71453818 IC50 = 52458 nM T91761 C49LMP 71455519 IC50 = 2180 nM T91761 C2R0KW 71455520 IC50 = 720 nM T91761 C7SX5M 71455521 IC50 = 1410 nM T91761 C6LH8Q 71455522 IC50 = 160 nM T91761 CL9YX8 71455523 IC50 = 10 nM T91761 C5B3VZ 71455524 IC50 > 100000 nM T91761 C9OZ7L 71455525 IC50 = 10324 nM T91761 CZE97Y 71455526 IC50 = 10068 nM T91761 CKT60L 71455860 Ki > 1500 nM T91761 C97EFZ 71457310 IC50 > 100000 nM T91761 C3ERY4 71457311 IC50 > 100000 nM T91761 CQBX94 71457312 IC50 = 130 nM T91761 CYIV59 71457313 IC50 = 4080 nM T91761 CM4XP7 71457314 IC50 > 100000 nM T91761 C7Y3CN 71457315 IC50 = 8341 nM T91761 CX9JD6 71457316 IC50 = 1045 nM T91761 COR7P9 71457317 IC50 = 22930 nM T91761 C6S2WH 71457340 IC50 = 21883 nM T91761 CNK30S 71459144 IC50 = 40 nM T91761 C2CMI9 71459145 IC50 = 5960 nM T91761 C7C5KR 71459146 IC50 = 73 nM T91761 CU6B3A 71459147 IC50 > 100000 nM T91761 CLN0C3 71459148 IC50 = 200 nM T91761 CS6JI3 71459149 IC50 = 1020 nM T91761 CKE8H3 71459150 IC50 = 2460 nM T91761 C4MA8X 71459191 IC50 = 20439 nM T91761 CLY18M 71460955 IC50 = 200 nM T91761 CQP21A 71460956 IC50 = 7570 nM T91761 CS3AW9 71460957 IC50 = 6645 nM T91761 C4LHT7 71462672 IC50 > 100000 nM T91761 CWD7E2 71462673 IC50 = 70 nM T91761 CX5K8Z 71462674 IC50 > 100000 nM T91761 C9FCM5 71462675 IC50 > 100000 nM T91761 CMF79G 71462676 IC50 = 21321 nM T91761 C8CG6H 71462712 IC50 = 9827 nM T91761 CEM84S 71462713 IC50 = 17744 nM T91761 CZM1K4 71765510 IC50 = 320 nM T91761 C98LKV 71777716 Ki = 8.4 nM T91761 C3MI4O 71777717 Ki = 0.7 nM T91761 C54XWG 72190869 IC50 > 10000 nM T91761 CS10DX 72544168 Ki = 1.9 nM T91761 CQH45K 72544389 Ki = 0.5 nM T91761 CVL5U1 72544390 Ki = 380 nM T91761 C2NV5Y 72544391 Ki = 2000 nM T91761 C21WYT 72544392 Ki = 230 nM T91761 CNOY69 72544393 Ki = 3500 nM T91761 CG38JZ 72544394 Ki = 50 nM T91761 CB9L0H 72544615 Ki = 85 nM T91761 C4OHT5 72544616 Ki = 3500 nM T91761 CA7C3K 72544617 Ki = 5.3 nM T91761 CJZV57 72544618 Ki = 6.6 nM T91761 CMS5O0 72544619 Ki = 2.5 nM T91761 CP7W1C 72544839 Ki = 30 nM T91761 CIE0T7 72544840 Ki = 1100 nM T91761 C0G4SO 72545063 Ki = 43 nM T91761 CFTK59 72705466 Ki > 10000 nM T91761 C1CU0H 72705467 Ki = 794.33 nM T91761 CX2AW3 72705468 Ki = 6.31 nM T91761 CVK4Z3 72705469 Ki = 501.19 nM T91761 C4ND6R 72705470 Ki = 63.1 nM T91761 CT67YO 72706106 Ki = 15.85 nM T91761 C9OQ2I 72710839 IC50 > 10000 nM T91761 C3L2WD 73292576 Ki = 5.3 nM T91761 C0P9LY 73292578 Ki = 10 nM T91761 CJ87SO 73292579 Ki = 75 nM T91761 CAS80Y 73292746 Ki = 8 nM T91761 C35BCQ 73292749 Ki = 37 nM T91761 C52LFH 73292907 Ki = 3 nM T91761 C0NE4O 73293422 Ki = 180 nM T91761 C26IVZ 73293424 Ki = 860 nM T91761 CIP49J 73293781 Ki < 0.1 nM T91761 CZ63BH 73293963 Ki = 42 nM T91761 CE1JT9 73294162 Ki = 0.3 nM T91761 C4FY5U 73346554 Ki = 0.3162 nM T91761 CPGD07 73348027 Ki = 3981.07 nM T91761 C05XEV 73348028 Ki = 158.49 nM T91761 CUW70Y 73348034 Ki = 0.3981 nM T91761 CFEU95 73348035 Ki = 15.85 nM T91761 C6K0UL 73348036 Ki > 10000 nM T91761 CD6KE7 73349574 Ki = 1.995 nM T91761 CV8UR4 73351136 Ki = 12.59 nM T91761 CAS60G 73352600 Ki = 3.981 nM T91761 CX75YR 73352604 Ki = 0.631 nM T91761 C5YKB4 73352605 Ki = 6.31 nM T91761 C03YUP 73355623 Ki = 19.95 nM T91761 C1A9PR 73357167 Ki = 1 nM T91761 CMEV76 74983355 Ki = 0.7 nM T91761 C0RP9Y 76309810 Ki = 0.6 nM T91761 C2A7SL 76320747 Ki = 6.4 nM T91761 CN39OQ 78341183 IC50 = 220 nM T91761 C1HW4B 89735655 IC50 = 4200 nM T91761 C5Q7UO 90036498 Ki = 31 nM T91761 C2ADJ1 90036634 Ki = 4000 nM T91761 CC06YJ 90036766 Ki = 22 nM T91761 CO51HL 90037453 Ki = 180 nM T91761 CX4C7W 90037556 Ki = 69 nM T91761 C6WQU2 90645540 Ki = 8.3 nM T91761 CSD73E 90645541 Ki = 0.8 nM T91761 C02KJP 90645542 Ki = 1.2 nM T91761 CE3OV2 90645543 Ki = 6.2 nM T91761 CY6L4N 90645544 Ki = 0.7 nM T91761 C7D5PI 90645545 Ki = 15 nM T91761 C93BGJ 90645546 Ki = 0.2 nM T91761 CSYV34 90656736 Ki = 3.4 nM T91761 C1CD8K 90656737 Ki = 1.7 nM T91761 C7C4KF 90656738 Ki > 4 nM T91761 CC6F3W 90656739 Ki = 53 nM T91761 CF89DA 90664659 IC50 = 22600 nM T91761 C64SIO 92042864 IC50 = 1070 nM T91761 C8HYU9 117926195 IC50 > 10000 nM T91761 CH4FU2 118641920 Ki = 0.27 nM T91761 C5EFI8 118641944 Ki = 14 nM T91761 CQ7Z0C 118641957 Ki = 8 nM T91761 CTP2E8 118737132 Ki = 0.5 nM T91761 C5GTM2 118737133 Ki = 0.2 nM T91761 C7MJ5H 118737134 Ki = 0.3 nM T91761 C3XF2A 118737135 Ki = 0.3 nM T91761 CNP5K8 118737136 Ki = 0.2 nM T91761 C8FDR1 118737137 Ki = 0.5 nM T91761 C37DUM 121293882 IC50 = 88 nM T91761 CXQR89 121294143 IC50 = 8.3 nM T91761 CFKD32 122191637 IC50 = 115 nM T91761 CLM7K3 122604539 IC50 > 10000 nM T91761 C01JHI 122604566 IC50 > 10000 nM T91761 CV89JM 132231876 IC50 = 23 nM T91761 C59HOQ 134277578 IC50 = 3.23 nM T91761 C0PZ5R 134277599 IC50 = 1.52 nM T91761 C7PWJ2 134277617 IC50 = 0.53 nM T91761 CRA2H1 134277633 IC50 = 1.5 nM T91761 CXJ8I0 134277643 IC50 = 0.34 nM T91761 C02RIA 134277647 IC50 = 0.67 nM T91761 CGH42R 134277652 IC50 = 0.72 nM T91761 COA14U 134277654 IC50 = 0.41 nM T91761 CQK0B5 134277685 IC50 = 10.1 nM T91761 C6S8VC 134277696 IC50 = 0.64 nM T91761 C49PIO 134277748 IC50 = 0.87 nM T91761 CD7VK4 134277767 IC50 = 1.62 nM T91761 CZ5E6L 134277773 IC50 = 0.7 nM T91761 C2CFK7 134277780 IC50 = 2.17 nM T91761 C6E7LW 134277790 IC50 = 0.81 nM T91761 C6T7NW 134277796 IC50 = 0.92 nM T91761 CU8ZP5 134277800 IC50 = 0.99 nM T91761 CTR4K6 134277828 IC50 = 0.58 nM T91761 C54FXD 134957362 IC50 > 10000 nM T91761 C6OE3V 135406885 IC50 = 160 nM T91761 COVY35 135406895 IC50 = 80 nM T91761 CUWM59 135409238 IC50 = 140 nM T91761 CG7K8I 135409247 IC50 = 170 nM T91761 CS0LR6 135445358 IC50 = 3980 nM T91761 CWM9Q1 135494486 IC50 = 350 nM T91761 C2U3AP 135514562 IC50 = 110 nM T91761 CK0M8W 135537103 IC50 = 250 nM T91761 CJ03PU 135566610 IC50 = 10.9 nM T91761 CQ9A5I 135566611 IC50 = 7 nM T91761 C42TOW 135566612 IC50 = 0.3 nM T91761 CN48IF 135566613 IC50 = 8.6 nM T91761 CIS2L5 135566617 IC50 = 150 nM T91761 C67IYS 135566618 IC50 = 1.9 nM T91761 CF48JM 135908497 IC50 = 560 nM T91761 C6H0AI 135957039 IC50 = 330 nM T91761 CP5SD0 136016241 IC50 = 2.4 nM T91761 CWB21F 136016374 IC50 = 2510 nM T91761 CCMG78 136016383 IC50 = 2000 nM T91761 CFTI43 136016384 IC50 = 1100 nM T91761 CBS87V 136016385 IC50 = 790 nM T91761 C05IWG 136016386 IC50 = 630 nM T91761 COPL16 136016393 IC50 = 630 nM T91761 C23APW 136016394 IC50 = 3160 nM T91761 C0XM8L 136016395 IC50 = 10000 nM T91761 CDS3A7 136016400 IC50 = 4360 nM T91761 CI37ET 136016401 IC50 = 1260 nM T91761 CD65WY 136016402 IC50 = 3160 nM T91761 CKWD23 136016403 IC50 = 1820 nM T91761 CO4C8Y 136016408 IC50 = 850 nM T91761 CUP47N 136016409 IC50 = 630 nM T91761 C4RMV8 136016410 IC50 = 1000 nM T91761 C0B7XQ 136016415 IC50 = 2060 nM T91761 C3Z6NG 136016416 IC50 = 1630 nM T91761 CXLZ12 136016417 IC50 = 2040 nM T91761 C9WVQ8 136016418 IC50 = 20400 nM T91761 C0MAS6 136016419 IC50 > 100000 nM T91761 C9BOX7 136016420 IC50 > 100000 nM T91761 C80OVA 136016421 IC50 = 630 nM T91761 C36PIS 136016422 IC50 = 500 nM T91761 CB8MI3 136016423 IC50 = 5000 nM T91761 CMY2N7 136016424 IC50 = 50100 nM T91761 CFY17E 136016425 IC50 = 1580 nM T91761 C7A9LY 136030592 IC50 = 120 nM T91761 CRA1H3 136030593 IC50 = 65 nM T91761 C4KLZ5 136030594 IC50 = 87 nM T91761 CVQF95 136030595 IC50 = 43 nM T91761 CRY2E5 136030598 IC50 = 140 nM T91761 CVZ3A4 136030599 IC50 = 260 nM T91761 C12OBR 136030600 IC50 = 70 nM T91761 C0Z7IM 136030629 IC50 = 20 nM T91761 CHMU19 136030633 IC50 = 110 nM T91761 CYRI63 136030634 IC50 = 100 nM T91761 CN3LU6 136030635 IC50 > 50000 nM T91761 C74LHJ 136030636 IC50 = 46 nM T91761 CFYO35 136030639 IC50 = 310 nM T91761 CP69FN 136030672 IC50 = 220 nM T91761 C6RIT2 136030673 IC50 > 50000 nM T91761 CF6D9C 136030674 IC50 = 66 nM T91761 CIC29X 136030675 IC50 = 120 nM T91761 CRY68L 136030705 IC50 = 190 nM T91761 C6Y0WA 136030710 IC50 = 370 nM T91761 CO4Z5H 136030736 IC50 = 67 nM T91761 C4S9QE 136030737 IC50 = 830 nM T91761 CPDZ24 136030738 IC50 = 45 nM T91761 C7GP4F 136030739 IC50 = 26 nM T91761 CLZ75U 136030740 IC50 = 85 nM T91761 CSA54K 136030741 IC50 = 730 nM T91761 C0TM4I 136030742 IC50 = 720 nM T91761 C4M9XD 136030743 IC50 = 10 nM T91761 CE9C0X 136030745 IC50 = 310 nM T91761 C1Z6KE 136030748 IC50 = 1500 nM T91761 C4U1ZE 136032568 IC50 = 240 nM T91761 CT3S7N 136032569 IC50 = 230 nM T91761 CO7BC1 136032578 IC50 = 22000 nM T91761 C5JM9H 136032600 IC50 = 80 nM T91761 C2JLY1 136032615 IC50 = 130 nM T91761 C0R9GU 136032627 IC50 = 90 nM T91761 CLR7S3 136059157 IC50 = 80 nM T91761 CUZ57E 136141542 IC50 = 2300 nM T91761 C9AT1U 136141543 IC50 = 98 nM T91761 CB74DR 136141544 IC50 = 900 nM T91761 C9PUM3 136141545 IC50 = 1410 nM T91761 C5YST1 136141546 IC50 = 750 nM T91761 CT6O7A 136141547 IC50 = 27 nM T91761 C71XIR 136141548 IC50 = 70 nM T91761 CK72XC 136141549 IC50 = 20 nM T91761 CS57KT 136141573 IC50 = 350 nM T91761 CNV86P 136141577 IC50 = 160 nM T91761 C5OW3D 136141585 IC50 = 530 nM T91761 C2AYS7 136141586 IC50 = 1000 nM T91761 C4C7OX 136141587 IC50 = 47 nM T91761 CYI26Q 136141588 IC50 = 72 nM T91761 C17KYN 136141589 IC50 = 1700 nM T91761 CY71KM 136141591 IC50 = 70 nM T91761 C7T0DC 136141592 IC50 = 1000 nM T91761 CLS79W 136141593 IC50 = 280 nM T91761 CZ7EX0 136183413 IC50 = 60 nM T91761 CQED29 136188798 IC50 = 140 nM T91761 CP5NE8 136188799 IC50 = 1600 nM T91761 CSRL54 136188800 IC50 = 36 nM T91761 C7VX4D 136188801 IC50 = 69 nM T91761 C9JS3P 136188802 IC50 = 250 nM T91761 CZ8IE1 136188803 IC50 = 340 nM T91761 CYLS64 136188804 IC50 = 300 nM T91761 CUE5X3 136188805 IC50 = 500 nM T91761 CU6Z0T 136188806 IC50 = 310 nM T91761 CJHT74 136188807 IC50 = 200 nM T91761 CTOR91 136188808 IC50 = 60 nM T91761 C9UIO6 136188809 IC50 = 110 nM T91761 CUI67Z 136188810 IC50 = 690 nM T91761 CUHP14 136188811 IC50 = 210 nM T91761 C9YLZ6 136188812 IC50 = 83 nM T91761 CPC8D4 136188813 IC50 = 780 nM T91761 C7TVJ9 136188814 IC50 = 860 nM T91761 C4AZP2 136188815 IC50 = 620 nM T91761 CI5V3P 136188816 IC50 = 1200 nM T91761 C28NFU 136188817 IC50 = 12000 nM T91761 C0BFO4 136188818 IC50 = 530 nM T91761 CB3IN0 136188819 IC50 = 16 nM T91761 CT9LV6 136188820 IC50 = 23 nM T91761 CD15JP 136188821 IC50 = 100 nM T91761 C9DU3V 136188822 IC50 = 100 nM T91761 CYZ9F4 136188823 IC50 = 990 nM T91761 CQL41E 136188824 IC50 = 260 nM T91761 CSH9W0 136188825 IC50 = 30 nM T91761 C1VJO0 136188826 IC50 = 77 nM T91761 C3UP6I 136188827 IC50 = 60 nM T91761 CW3E2V 136188828 IC50 = 130 nM T91761 CW1IV2 136199382 IC50 = 120 nM T91761 CJ0FZ4 136199383 IC50 = 190 nM T91761 CE27WO 136199384 IC50 = 80 nM T91761 C5Q0ZC 136199385 IC50 = 310 nM T91761 CB58FG 136199386 IC50 = 140 nM T91761 CTY4Q1 136199387 IC50 = 70 nM T91761 CY4TS0 136199388 IC50 = 200 nM T91761 C8EC0L 136199389 IC50 = 280 nM T91761 CSKP13 136199390 IC50 = 27000 nM T91761 CU8P2N 136199391 IC50 = 300 nM T91761 CRHS39 136199392 IC50 = 70 nM T91761 C26NEM 136254164 IC50 = 200 nM T91761 CXC69T 137321158 IC50 = 60 nM T91761 C3Z4AT 137321159 IC50 > 10000 nM T91761 C7TG3J 137641313 IC50 > 19952.62 nM T91761 C4DRX1 137643187 IC50 = 2190 nM T91761 C28QUP 137652864 IC50 = 5655 nM T91761 CRWA29 139030520 IC50 = 306.9 nM T91761 C9ZYG8 141366083 IC50 = 290 nM T91761 C4OD9Q 145967187 IC50 = 15.1 nM T91761 CE31VG 145979714 IC50 > 10000 nM T91761 C9BX4U 145988956 IC50 > 10000 nM T91761 C2MD1Q 155513187 IC50 > 10000 nM T91761 CA7O4B 155513491 IC50 = 5.4 nM T91761 C7AMX8 155514903 IC50 = 3.6 nM T91761 CI23DH 155516489 IC50 = 3.7 nM T91761 CU0VL1 155517584 IC50 = 22 nM T91761 C3NA2I 155519537 IC50 > 1000 nM T91761 CRT67D 155526236 IC50 = 1.3 nM T91761 CRC38Y 155526544 IC50 = 87 nM T91761 CE3OH1 155527121 IC50 < 1.26 nM T91761 CUXA18 155529935 IC50 = 2.3 nM T91761 CL0US4 155530459 IC50 = 0.5 nM T91761 C2WCU6 155530774 IC50 = 5.4 nM T91761 C1NGV5 155534208 IC50 = 3.7 nM T91761 C1UJ4T 155534213 IC50 = 32 nM T91761 CU9S7B 155535315 IC50 = 4.8 nM T91761 CBZ4V6 155536645 IC50 = 1437 nM T91761 C2CG1A 155537016 IC50 > 10000 nM T91761 C0JL6C 155537712 IC50 = 23 nM T91761 CWY1O0 155538122 IC50 > 10000 nM T91761 CJ5OI0 155541008 IC50 = 423 nM T91761 CH10DU 155542091 IC50 = 5.1 nM T91761 CELG50 155543350 IC50 = 469 nM T91761 CW73EO 155543439 IC50 < 1.26 nM T91761 CO1S0E 155546265 IC50 = 42 nM T91761 C2ZHA0 155547912 IC50 = 22 nM T91761 C0C1FI 155548702 IC50 = 126 nM T91761 C79PYG 155550586 IC50 = 15 nM T91761 C6YE8Z 155552072 IC50 = 2133 nM T91761 CXB6U7 155552682 IC50 = 14 nM T91761 C0HUL3 155552710 IC50 = 7.8 nM T91761 CZ9OW5 155558028 IC50 = 14 nM T91761 CPAV79 155559005 IC50 = 55 nM T91761 C4L6HQ 155559509 IC50 = 375 nM T91761 C51IBQ 155560019 IC50 = 7.1 nM T91761 C61NVM 155560973 IC50 = 75 nM T91761 CAC85T 155564156 IC50 = 74 nM T91761 CDAY91 155568779 IC50 = 12 nM T91761 CC29WQ 155568870 IC50 > 10000 nM T91761 CGU74Q 155569301 IC50 = 2.2 nM T91761 D00ERW 44444843 Ki > 1525 nM T91761 D00HVA 11624601 Ki > 3800 nM T91761 D01RHR 71519693 IC50 > 30000 nM T91761 D01VFR 4708 IC50 > 30000 nM T91761 D04PEI 11467730 Ki = 16 nM T91761 D05RPN 11527400 IC50 = 96 nM T91761 D06BJG 71556703 IC50 > 30000 nM T91761 D06WGX 9549184 IC50 > 25000 nM T91761 D0D6MH 11617559 IC50 > 16000 nM T91761 D0E7VO 59627005 IC50 = 72.2 nM T91761 D0GN5Z 5281295 IC50 = 2020 nM T91761 D0J3LR 11634725 Ki > 4000 nM T91761 D0OZ2S 11785878 IC50 > 20000 nM T91761 D0Q0YV 24944925 IC50 = 5495.41 nM T91761 D0Q3NG 11715520 Ki > 3800 nM T91761 D0S7IE 11658882 Ki > 3800 nM T54132 D0S6QR 214350 EC50 = 2400 nM T54132 D0X7GL 121892 EC50 = 3900 nM T54132 C30IVC 155491024 EC50 = 10500 nM T54132 CTJ34I 155491025 EC50 = 920 nM T54132 D0FF6S 16038374 IC50 > 10000 nM T77139 D0E3TC 44259 IC50 = 10.9 nM T77139 C3VRO9 44557921 IC50 > 10000 nM T77139 CV63UL 67240318 IC50 > 10000 nM T77139 C6VB3O 145925651 IC50 >= 5000 nM T77139 C2MD1Q 155513187 IC50 > 10000 nM T77139 D0J3LR 11634725 Ki > 4000 nM T37693 D07ILQ 4671 Ki > 5000 nM T37693 D0E6YQ 1935 Ki > 1000 nM T37693 D0L7AS 5284592 Ki = 1.84 nM T37693 D0O1UZ 644019 Ki = 372 nM T37693 D0O3OS 104850 Ki = 1.1 nM T37693 D0P1FO 16078 EC50 = 1.5 nM T37693 D0R1RS 3715 Ki > 20000 nM T37693 D0T9TJ 3034010 Ki > 10000 nM T37693 D0U5CE 1548943 Ki > 10000 nM T37693 D08DGC 3083542 Ki = 170.5 nM T37693 D0I4PW 60164925 EC50 = 6.2 nM T37693 D0J6KZ 57331749 IC50 = 24 nM T37693 D0Q7NB 10253143 EC50 = 50 nM T37693 D0Q8WG 67029278 EC50 = 0.61 nM T37693 D0U2BH 65064 Ki = 42800 nM T37693 D0W3GL 9849616 Ki = 442 nM T37693 D0Y9RO 107778 Ki = 0.15 nM T37693 D00GES 66553204 IC50 > 1000 nM T37693 D01RIT 24857045 IC50 = 3838.3 nM T37693 D02TOI 121231416 EC50 = 0.3 nM T37693 D02ZVY 72712999 Ki = 426 nM T37693 D07BFP 60148509 Ki = 134 nM T37693 D07IHT 4296438 EC50 = 159.1 nM T37693 D07NAA 24945235 IC50 > 10000 nM T37693 D07ULI 5752181 EC50 = 296 nM T37693 D09GJQ 73330476 Ki = 0.8 nM T37693 D0D1EI 72713196 Ki = 1046 nM T37693 D0DE0C 72713199 Ki = 60.2 nM T37693 D0E6YT 71539748 EC50 = 19 nM T37693 D0FS0D 44571565 IC50 > 10 nM T37693 D0GQ8W 46871948 Ki = 7.5 nM T37693 D0GX6V 23624319 Ki = 804 nM T37693 D0I1XE 72713197 Ki = 2360 nM T37693 D0J5XM 25098114 IC50 = 5200 nM T37693 D0JW7T 9868408 Ki = 1110 nM T37693 D0KD5X 44247611 IC50 = 636 nM T37693 D0KX2W 46889224 Ki > 1000 nM T37693 D0M2RT 24863732 Ki = 398 nM T37693 D0O4RN 24744027 IC50 > 10000 nM T37693 D0TI3Q 11555526 Ki > 10000 nM T37693 D0V0UW 25098092 IC50 = 3800 nM T37693 D0WJ3F 71584280 Ki = 0.5 nM T37693 D0YZ8I 4273754 Ki = 13.3 nM T37693 D0Z8WF 24944528 IC50 = 19000 nM T37693 D03ACT 9844711 Ki = 22.7 nM T37693 D06TGE 11226090 Ki = 290 nM T37693 D0A9OR 11179267 Ki > 1000 nM T37693 D0H1FL 11316919 Ki > 10000 nM T37693 D0J0AE 10052040 Ki = 7700 nM T37693 D0J7RW 5311501 Ki = 0.28 nM T37693 C1S7VI 2415 Ki = 435 nM T37693 C5H9CN 9287 Ki > 10000 nM T37693 CQP80E 15339 Ki = 4021 nM T37693 C9WJ7H 25957 Ki = 960 nM T37693 C3ERF2 30219 Ki = 257 nM T37693 CWYV98 39860 Ki = 6.31 nM T37693 CTK25Q 72277 Ki = 361300 nM T37693 C8SD5O 72300 Ki = 1440 nM T37693 C0AGE7 78262 Ki > 10000 nM T37693 CJ5T2N 98523 Ki = 56 nM T37693 C0QSW4 104849 Ki = 1580 nM T37693 CNIW58 107905 Ki = 95600 nM T37693 CR4JB5 129128 Ki = 2.9 nM T37693 CRYZ13 169652 Ki = 88 nM T37693 CMP4K1 192007 Ki = 2143 nM T37693 C4P1GV 194130 Ki = 9 nM T37693 C3T5KU 292955 Ki > 10000 nM T37693 CVL1A0 320263 Ki > 10000 nM T37693 CL3UD5 320264 Ki > 10000 nM T37693 C0TJF6 321643 Ki = 192 nM T37693 C94GYM 331257 EC50 = 1200 nM T37693 CFY02L 356017 Ki > 10000 nM T37693 C8X7ST 356018 Ki > 10000 nM T37693 C5V0SH 386338 Ki = 400 nM T37693 C8LY2I 391240 Ki = 1993.94 nM T37693 CE7NH5 470766 EC50 = 980 nM T37693 CJ3NQ1 601368 Ki = 2060 nM T37693 CU57BO 601392 IC50 > 10000 nM T37693 C37RCW 622545 EC50 = 4780 nM T37693 CPK8U9 695120 Ki > 10000 nM T37693 CZ9SJ1 695133 Ki > 10000 nM T37693 CECS97 708647 Ki > 10000 nM T37693 CP64YR 727029 EC50 = 7943.28 nM T37693 CGT6F3 738959 Ki > 10000 nM T37693 CMR9E1 746182 Ki = 700 nM T37693 CT7DE5 759445 Ki = 660 nM T37693 CR8WV7 834671 Ki = 6741 nM T37693 C3VXW6 836750 Ki > 10000 nM T37693 CDE0L5 853260 EC50 = 199 nM T37693 C90NZF 853261 EC50 = 24.8 nM T37693 CV24TH 868829 Ki = 495.77 nM T37693 CVRG42 872331 Ki > 10000 nM T37693 CQ3K8M 897320 Ki = 621 nM T37693 C7SQL6 900707 Ki > 10000 nM T37693 COU5J2 900710 Ki > 10000 nM T37693 C6D7XU 991033 Ki = 783 nM T37693 C6O3XR 991035 Ki = 10899.99 nM T37693 C1L2CV 1000896 Ki = 1.35 nM T37693 C6SDA3 1001644 Ki = 2400 nM T37693 CB79QJ 1034762 Ki = 16.8 nM T37693 CTXK08 1040500 Ki = 1785.22 nM T37693 CS39EC 1068516 EC50 = 14 nM T37693 CFY2M3 1075977 Ki = 1866 nM T37693 CZR2G8 1098594 Ki = 111.87 nM T37693 C4NL1G 1127069 Ki = 360 nM T37693 C1GSP2 1144102 EC50 = 139 nM T37693 C8O0RS 1202067 IC50 = 4.2 nM T37693 CZY91E 1216383 EC50 = 27 nM T37693 C0MYU2 1281700 Ki > 10000 nM T37693 C8KD9F 1281702 Ki > 10000 nM T37693 CH8PY0 1281704 Ki > 10000 nM T37693 CX5F6G 1281706 Ki > 10000 nM T37693 C1ZS6H 1340631 Ki > 20000 nM T37693 CM2D5Q 1350471 EC50 = 10 nM T37693 CH5TO8 1581054 Ki = 19.3 nM T37693 C7UPS9 1602258 Ki < 25 nM T37693 C3CZ0N 1626958 Ki = 18.5 nM T37693 CF57VU 1649385 Ki = 59.81 nM T37693 CZ71FX 1722112 Ki > 10000 nM T37693 CT42LA 1837112 Ki = 2.1 nM T37693 C8Z0YQ 1895552 Ki < 1000 nM T37693 C6F1EP 2084332 EC50 = 184 nM T37693 CC0Y2N 2086721 EC50 = 44.4 nM T37693 C3WIV0 2117799 Ki = 1300 nM T37693 CU50TE 2174064 EC50 = 21 nM T37693 CM4S0X 2188265 Ki < 25 nM T37693 C5B6FD 2317892 EC50 = 8 nM T37693 CIT03M 2323038 Ki > 10000 nM T37693 CL85HP 2526892 Ki = 2226 nM T37693 C38NEA 2599179 EC50 = 154 nM T37693 CV8SL5 2599466 EC50 = 21 nM T37693 CF16MC 2600862 EC50 = 5 nM T37693 COM7R5 2623606 EC50 = 3 nM T37693 C3Z7OT 2666218 EC50 = 14100 nM T37693 C62SYO 2691386 EC50 = 240 nM T37693 C95VEI 2729564 IC50 > 10000 nM T37693 CO04GZ 2787166 EC50 > 10000 nM T37693 CIUG12 2787170 EC50 = 15 nM T37693 CYG2A9 2801231 EC50 = 3 nM T37693 CFV1D2 2808251 EC50 = 630 nM T37693 CUZ19I 2825619 EC50 = 5011.87 nM T37693 CBAE76 2825620 EC50 = 5011.87 nM T37693 C85HRJ 2836420 Ki > 10000 nM T37693 CSEB28 2836426 EC50 = 100 nM T37693 CDTK31 2846758 Ki = 2.15 nM T37693 C7SD1X 2850042 Ki = 5.08 nM T37693 C9JT7I 2851184 EC50 = 55 nM T37693 C9HCD2 2853642 Ki = 2.46 nM T37693 CI04TU 2987572 EC50 > 10000 nM T37693 C1Q9NO 3042143 IC50 > 1000 nM T37693 C86NOR 3082311 Ki = 26.6 nM T37693 C5MKT8 3168799 Ki < 25 nM T37693 C8KH0Z 3258886 Ki > 10000 nM T37693 CE24BQ 3298404 Ki = 244.06 nM T37693 CQ38BO 3340785 Ki = 4900 nM T37693 CLCV10 3372949 Ki > 10000 nM T37693 CSU8B7 3379236 Ki = 17400 nM T37693 CCQZ29 3426415 Ki = 10000 nM T37693 C2C9PX 3579176 EC50 = 23 nM T37693 CQT7K2 3580670 EC50 > 20000 nM T37693 C08PSA 3643741 Ki > 10000 nM T37693 CTS89I 3703767 Ki = 58 nM T37693 CA1O6R 3868445 IC50 > 10000 nM T37693 C8O1VI 3929482 EC50 < 1 nM T37693 CJ2D3A 3932001 Ki = 1069 nM T37693 CIJ95Y 4055807 Ki = 3100 nM T37693 C5OVS7 4140053 EC50 = 600 nM T37693 CM31EP 4262768 EC50 = 131.1 nM T37693 C6K2SR 4346308 Ki = 10000 nM T37693 C18UZB 4382038 EC50 = 154 nM T37693 C5IJ2F 4458788 EC50 = 500 nM T37693 CGO5X8 4478978 Ki = 1500 nM T37693 CFYQ35 4489585 Ki = 35330 nM T37693 CXC9U2 4554609 Ki > 10000 nM T37693 CBC0D2 4559116 Ki = 9.24 nM T37693 C5PA1K 4621779 Ki = 9400 nM T37693 CUCD57 4693614 Ki = 10000 nM T37693 C8YL3A 4722382 Ki = 19950 nM T37693 CO0EK1 4736636 Ki = 3919 nM T37693 CX2GY3 4790042 EC50 = 195 nM T37693 C56SGI 4963989 Ki > 10000 nM T37693 C0LK2Z 4996150 Ki = 4953 nM T37693 CVQR47 5030390 EC50 = 200.7 nM T37693 CX46YD 5164405 Ki = 35 nM T37693 CF3KG6 5281515 Ki = 150 nM T37693 C3J9NW 5285645 EC50 = 10000 nM T37693 CMV9I2 5290645 EC50 > 3000 nM T37693 COT13X 5292590 EC50 > 3000 nM T37693 C9SC1F 5311172 Ki = 11.2 nM T37693 CZ46HG 5315659 Ki = 153 nM T37693 CK0X9M 5318518 EC50 = 41.7 nM T37693 C47FZC 5319201 Ki > 10000 nM T37693 CIU1J6 5321844 IC50 = 2 nM T37693 CJI57N 5321851 EC50 = 170 nM T37693 CPFC04 5368482 Ki > 40000 nM T37693 CX1RJ0 5376147 EC50 > 3000 nM T37693 CZ8NS2 5714946 EC50 > 3000 nM T37693 C09MQY 5714954 EC50 > 3000 nM T37693 CZ31XM 5722610 EC50 = 110 nM T37693 CY87CV 5730854 EC50 > 3000 nM T37693 CC4B0K 5917569 Ki > 10000 nM T37693 CC6G3O 6401050 EC50 = 617 nM T37693 C0JQ4U 6401059 EC50 = 112 nM T37693 C4NI8E 6409200 EC50 = 2185 nM T37693 C3RNJ8 6434324 IC50 = 19900 nM T37693 CH97NY 6440539 Ki = 9044 nM T37693 CWF02M 6440803 Ki = 3140 nM T37693 CF2B7X 6442405 Ki = 38300 nM T37693 C4WPT9 6453891 Ki = 51 nM T37693 C3TLF8 6481606 Ki > 10000 nM T37693 CPLC65 6481633 Ki > 10000 nM T37693 C2C4KE 6604176 Ki = 2.1 nM T37693 CP6RW5 6621153 Ki = 22800 nM T37693 C1ZW6X 6973727 IC50 = 45 nM T37693 CRWD27 7620138 Ki = 31 nM T37693 CDUC94 7620149 Ki = 22 nM T37693 CO3M5A 7620714 Ki = 2.2 nM T37693 C16AMB 7620725 Ki = 0.7 nM T37693 C7H2FT 7929121 Ki = 170 nM T37693 C8POQ0 7929124 Ki = 2900 nM T37693 C45OEP 8178387 Ki = 5.6 nM T37693 CPM3X1 8712703 Ki = 19 nM T37693 CUPW49 8803123 EC50 = 3 nM T37693 C67QOU 8803155 EC50 = 1 nM T37693 CL3DG9 8916493 EC50 = 33 nM T37693 C8E0JX 8916569 EC50 = 6450 nM T37693 C7I8PY 9123860 Ki > 10000 nM T37693 CGFY81 9123866 Ki > 10000 nM T37693 CQ3S9L 9124038 Ki > 10000 nM T37693 CZLT78 9192580 Ki > 10000 nM T37693 C2INQ1 9295948 EC50 > 20000 nM T37693 CLI69S 9314544 EC50 = 82 nM T37693 C32SMR 9401432 Ki > 10000 nM T37693 CH0V2X 9456049 Ki > 10000 nM T37693 CVZG73 9799417 Ki = 19 nM T37693 CTA5Z1 9800032 Ki = 1.6 nM T37693 C9V2CG 9800960 Ki = 4.07 nM T37693 CST19C 9801139 Ki > 1000 nM T37693 CNV3H9 9817492 Ki = 0.032 nM T37693 C8MS1D 9821406 Ki > 1000 nM T37693 CWGT52 9825614 EC50 = 2.3 nM T37693 CVR42O 9826744 IC50 = 1100 nM T37693 CUL5C1 9828471 IC50 = 3.5 nM T37693 CU96OX 9829238 Ki = 11 nM T37693 COD3T8 9829239 Ki = 8 nM T37693 C94AQK 9840457 IC50 > 10000 nM T37693 CRM5P4 9845561 Ki = 234422881.5 nM T37693 C73YBV 9866977 IC50 = 3.162 nM T37693 CQWX41 9867382 Ki = 1.05 nM T37693 C9Q2UN 9867770 Ki = 0.087 nM T37693 CRP37G 9868656 IC50 = 610 nM T37693 CG17YV 9881987 Ki = 54 nM T37693 CSM14G 9883343 Ki = 51.5 nM T37693 C1RO9M 9887568 Ki = 2240 nM T37693 CJG8R5 9888694 Ki = 0.019 nM T37693 C8H1QX 9908345 Ki = 13000 nM T37693 C3ND1I 9908916 Ki = 1.099 nM T37693 CB4L7I 9911463 EC50 = 0.65 nM T37693 C95PSM 9912393 Ki = 4668 nM T37693 CT4GD0 9914194 Ki = 1.8 nM T37693 CA4W6I 9931203 EC50 = 245 nM T37693 CF92JW 9935463 IC50 = 440 nM T37693 CLU0R5 9949177 Ki = 2.3 nM T37693 CI8F4E 9952038 Ki = 8.5 nM T37693 CJLB98 9953325 Ki = 0.01 nM T37693 C7BXH9 9956047 Ki = 1 nM T37693 CXF43E 9956414 Ki = 28000 nM T37693 C9LYH8 9975456 Ki = 0.39 nM T37693 C07RPH 9976253 Ki = 2.72 nM T37693 C5CA4N 9978707 EC50 = 250 nM T37693 CBKD01 9980724 EC50 = 10000 nM T37693 CG56EX 10002881 EC50 = 220 nM T37693 C5B0KC 10002952 Ki = 0.52 nM T37693 C92WBO 10024336 EC50 = 126 nM T37693 C5TRX2 10025406 EC50 = 63 nM T37693 CXQ29Y 10028229 IC50 = 5400 nM T37693 CA06TQ 10028888 IC50 = 5400 nM T37693 C6EML8 10029316 IC50 = 1970 nM T37693 CGNA89 10045603 EC50 = 40 nM T37693 CPI2Q0 10049358 EC50 = 33 nM T37693 CRSZ23 10051574 Ki = 9 nM T37693 CSOR04 10070428 EC50 = 50 nM T37693 C5B4HJ 10071498 EC50 = 125 nM T37693 C6R1ZC 10071974 EC50 = 1580 nM T37693 C29SQA 10073313 EC50 = 79.43 nM T37693 CB34HN 10084135 IC50 = 59 nM T37693 CVDZ53 10088884 Ki = 55.3 nM T37693 C6CB0K 10091328 Ki = 5.4 nM T37693 C3SGD4 10091426 Ki = 50 nM T37693 CRKT12 10092198 EC50 = 455 nM T37693 CZ5F8M 10094322 EC50 = 63.1 nM T37693 CI7X0M 10095319 EC50 = 230 nM T37693 CETX82 10097960 Ki > 10000 nM T37693 CF2ZS1 10099858 Ki = 0.7 nM T37693 C9WJ0K 10110855 Ki > 1000 nM T37693 C5TH1Q 10112572 Ki = 6300 nM T37693 C46EPR 10113020 Ki = 2960 nM T37693 C27MKW 10114327 Ki > 1000 nM T37693 C2W7ET 10127144 IC50 = 310 nM T37693 CRZ04L 10127496 Ki = 357 nM T37693 C2BAG9 10135518 Ki > 1000 nM T37693 C9XQ1F 10136173 Ki = 3082 nM T37693 CO9KZ4 10140173 Ki = 2700 nM T37693 C4VC9R 10141881 Ki = 2700 nM T37693 C3Q9WV 10151871 IC50 = 2300 nM T37693 CFI4R1 10152346 IC50 = 450 nM T37693 C0O2NM 10153212 Ki = 0.39 nM T37693 CN9Q6F 10157610 Ki = 70 nM T37693 CU5JQ8 10159384 Ki = 77 nM T37693 CPAX61 10159759 Ki = 5300 nM T37693 C42WGZ 10174045 Ki = 9 nM T37693 CLP8Z2 10174286 IC50 = 4100 nM T37693 C5XWL2 10175260 Ki = 0.38 nM T37693 C2QE6Z 10186399 Ki = 2312 nM T37693 CY4EQ6 10195058 IC50 = 730 nM T37693 CS49KR 10195276 IC50 = 1700 nM T37693 CRDN48 10195347 Ki = 160 nM T37693 CS1V9E 10195397 Ki = 3297 nM T37693 CS2O5P 10195715 IC50 = 4100 nM T37693 CY4O5A 10195774 IC50 = 1100 nM T37693 CV1NH0 10199993 Ki = 67 nM T37693 C5UFP0 10200053 Ki = 118.6 nM T37693 CST52D 10200054 Ki > 1000 nM T37693 CCF80H 10216046 Ki = 0.8 nM T37693 CD3M8S 10216984 Ki = 774 nM T37693 CGD2O6 10218033 IC50 = 5600 nM T37693 CDF3J9 10220912 IC50 = 131 nM T37693 C3RAT1 10221835 Ki > 1000 nM T37693 CZ5S1P 10224082 Ki = 1900 nM T37693 CSYH78 10225801 Ki = 250 nM T37693 C51GDE 10227614 Ki = 8 nM T37693 CZ4XV5 10249485 EC50 = 2 nM T37693 CL3C6O 10250275 Ki = 14 nM T37693 C4I8EY 10250508 EC50 = 200 nM T37693 C5RHE4 10252734 Ki = 0.037 nM T37693 C9JZ2C 10253141 EC50 = 630 nM T37693 C03DKF 10253142 EC50 = 100 nM T37693 CUF43P 10254284 IC50 = 440 nM T37693 CQ8AX2 10257665 Ki = 8 nM T37693 C8YH0U 10271378 Ki > 1000 nM T37693 CZN0M8 10271619 Ki > 1000 nM T37693 CKY63T 10272277 Ki > 1000 nM T37693 CX25NI 10276190 Ki = 2300 nM T37693 CW65AL 10277824 Ki = 12 nM T37693 CM86TS 10287827 IC50 = 860 nM T37693 CD3BM8 10289976 Ki = 7.6 nM T37693 CS3L9E 10294441 Ki > 1000 nM T37693 CU45SK 10294778 Ki = 133 nM T37693 CQR29X 10297613 Ki = 542 nM T37693 COE0K9 10310644 IC50 = 430 nM T37693 C35JNY 10310812 IC50 = 4400 nM T37693 CG3M2Y 10310945 IC50 = 465 nM T37693 C78QAR 10311022 IC50 = 3800 nM T37693 CE4HG6 10311095 IC50 = 5200 nM T37693 C08NME 10311098 IC50 = 4200 nM T37693 CRP35L 10311846 IC50 = 820 nM T37693 CHOT95 10312127 Ki = 5.5 nM T37693 C8F1LK 10318708 EC50 = 80 nM T37693 C27TCH 10319351 Ki = 3.981 nM T37693 CI20DM 10324989 Ki = 0.4 nM T37693 COU9I0 10340138 Ki = 0.52 nM T37693 C4AJ0X 10341839 EC50 = 125 nM T37693 CFXA48 10343679 EC50 = 49 nM T37693 C06HBC 10343680 EC50 = 80 nM T37693 C6F7DJ 10346347 EC50 = 2 nM T37693 C7SW3C 10360860 Ki = 2.897 nM T37693 CDR50J 10361702 Ki = 0.8511 nM T37693 CW9P2U 10364379 EC50 = 80 nM T37693 CZ1CH4 10365766 EC50 = 25000 nM T37693 CI2MZ3 10366006 IC50 = 2100 nM T37693 CLVC49 10367110 Ki = 228 nM T37693 C5QT1A 10367921 IC50 > 2000 nM T37693 CD6MC9 10382701 Ki = 2.897 nM T37693 C7HV9R 10383130 Ki = 23.6 nM T37693 CJ4NL2 10385575 EC50 = 125.89 nM T37693 CIK8N3 10386267 EC50 = 8.7 nM T37693 CVM7O3 10386369 EC50 = 158 nM T37693 CM1C5I 10407577 Ki = 0.22 nM T37693 C9Y3TJ 10410512 IC50 = 1000 nM T37693 C8K7VS 10410589 EC50 = 125 nM T37693 CHK4R7 10413523 IC50 = 3400 nM T37693 C7JWT4 10415499 Ki = 0.9 nM T37693 CEG3A8 10430464 EC50 = 310 nM T37693 CI39ZO 10433670 IC50 = 360 nM T37693 CO1GI7 10435654 Ki = 20 nM T37693 CFWR83 10449945 Ki = 2 nM T37693 CA9EN5 10453633 Ki = 0.2 nM T37693 C3YH6T 10453719 EC50 = 465 nM T37693 C97LHV 10454092 EC50 = 50 nM T37693 C09LYS 10455714 EC50 = 214 nM T37693 C2JX0C 10456931 IC50 = 640 nM T37693 C73TBN 10468802 Ki > 10000 nM T37693 C5BIY8 10471670 Ki = 9.8 nM T37693 CV1S8R 10478331 IC50 = 1900 nM T37693 CDIQ59 10478467 EC50 = 400 nM T37693 CCEA61 10479060 Ki = 45.5 nM T37693 CW0K3P 10479686 Ki = 5841 nM T37693 CY5Q3L 10500128 Ki = 0.2 nM T37693 CY1Z0O 10500863 Ki = 276 nM T37693 C3HE0R 10522112 Ki = 3.3 nM T37693 CH1NY0 10527931 Ki = 1.1 nM T37693 CLZ9Q7 10545949 Ki = 611 nM T37693 CZ67QE 10546891 Ki = 1 nM T37693 C2YTM0 10546947 Ki = 132 nM T37693 C3BU8K 10547208 Ki = 12.39 nM T37693 CN6CJ9 10566956 Ki = 113 nM T37693 CB8L6S 10577158 Ki > 10000 nM T37693 C4WX2N 10596625 Ki > 10000 nM T37693 CEF0Y9 10597702 Ki = 3.8 nM T37693 C7Q6NW 10618930 EC50 = 0.79 nM T37693 CLE3D5 10619854 Ki = 2.05 nM T37693 CWI98J 10620782 Ki = 4.8 nM T37693 CQG23I 10639725 Ki = 6 nM T37693 CP07NE 10642025 Ki = 83.18 nM T37693 CNE1B0 10647307 Ki > 10000 nM T37693 C40THY 10667130 Ki = 100 nM T37693 CLU8K3 10667559 Ki = 658 nM T37693 CN0IJ1 10673015 Ki > 10000 nM T37693 C6C4KH 10687450 Ki = 67 nM T37693 C1W3QS 10713019 Ki = 3 nM T37693 CE8Q6I 10720372 Ki = 441.7 nM T37693 CDNT67 10721387 Ki > 10000 nM T37693 CHN83D 10738579 Ki = 286 nM T37693 CLA8R7 10765468 Ki = 17.3 nM T37693 C1GYK3 10766696 Ki = 3.2 nM T37693 C2EPG7 10784206 EC50 = 4.6 nM T37693 CI71YU 10789819 Ki = 214 nM T37693 C7WKY6 10807814 Ki = 167 nM T37693 C6XQA9 10812269 Ki = 529 nM T37693 C8WSJ0 10831231 Ki = 31.99 nM T37693 CRI9J2 10833730 Ki = 2.9 nM T37693 C8LF3D 10858553 Ki > 10000 nM T37693 C3TC7H 10871668 Ki > 10000 nM T37693 CYZ85H 10883832 Ki > 1000 nM T37693 CWGU04 10884669 Ki = 1250 nM T37693 C2NEC5 10894571 Ki = 7820 nM T37693 CK8MY5 10895601 Ki = 67 nM T37693 CSG5H6 10902223 Ki > 10000 nM T37693 C1Q6BG 10906799 Ki = 146 nM T37693 CSR89T 10917163 Ki = 5900 nM T37693 C5BL2J 10928080 Ki > 1000 nM T37693 C8SL5H 10928335 Ki = 2 nM T37693 CQJS43 10928493 Ki = 2850 nM T37693 C8WA9L 10949701 Ki > 1000 nM T37693 CKT6I1 10950375 Ki = 3.6 nM T37693 C52ZOA 10961413 Ki = 5720 nM T37693 CB9M5P 10971904 Ki = 1740 nM T37693 CS30GQ 10972649 Ki = 6870 nM T37693 CK6O4D 10972872 Ki = 257 nM T37693 CYHU13 10973077 Ki > 1000 nM T37693 CKX4U3 10982154 Ki = 12100 nM T37693 C2XHD6 10982174 Ki = 1.905 nM T37693 CCU7E9 10983017 Ki = 1770 nM T37693 CY2X8K 11003836 Ki = 400 nM T37693 C0AS5E 11015192 Ki > 5000 nM T37693 CIY7D6 11037300 Ki = 4270 nM T37693 CCI2L6 11045217 Ki > 10000 nM T37693 C1S7MK 11048823 Ki = 19.5 nM T37693 CMIK78 11049238 Ki = 69 nM T37693 CV37YF 11057719 Ki > 1000 nM T37693 CHN0G5 11058423 Ki > 5000 nM T37693 CQ5A6M 11070648 Ki = 2400 nM T37693 CI8A6B 11076506 Ki > 10000 nM T37693 C92DRC 11080633 Ki = 2620 nM T37693 CH7VZ1 11090651 Ki > 1000 nM T37693 CYSC34 11090957 Ki > 1000 nM T37693 C6BM2P 11101378 Ki > 5000 nM T37693 C1YE9J 11102012 Ki > 1000 nM T37693 C3PGJ1 11102177 Ki = 1600 nM T37693 CDUO30 11103143 Ki = 28.1 nM T37693 CFP16U 11122439 Ki = 6660 nM T37693 CPK63M 11133144 Ki > 5000 nM T37693 CG03AU 11133899 Ki = 704 nM T37693 C63VBU 11143777 Ki > 1000 nM T37693 CJ8ED4 11152088 Ki = 79.98 nM T37693 C9E2AP 11152300 Ki > 10000 nM T37693 CA79PI 11153626 Ki = 0.1 nM T37693 CB47FY 11154357 EC50 = 79.43 nM T37693 CA5OX2 11154964 IC50 = 5.012 nM T37693 CTN10X 11155520 Ki = 758 nM T37693 CS92VB 11167681 IC50 = 1500 nM T37693 CAP2S3 11168529 Ki = 746 nM T37693 CGW7M1 11176619 Ki = 10.99 nM T37693 CW8V3S 11179949 Ki = 3515 nM T37693 CJ9U8Q 11185771 Ki > 10000 nM T37693 C92AOP 11187538 Ki > 10000 nM T37693 CT8XE9 11188464 Ki = 8.9 nM T37693 CEST31 11188528 Ki = 76 nM T37693 CRK7V9 11189799 Ki = 2520 nM T37693 C9E3HK 11190290 Ki > 10000 nM T37693 C7VB3Y 11190694 Ki = 1590 nM T37693 CM41GW 11192215 IC50 = 1800 nM T37693 C59LVQ 11199737 EC50 = 794.33 nM T37693 CNF70Q 11201613 Ki = 0.3981 nM T37693 CMXO58 11202164 Ki > 10000 nM T37693 CB06ZT 11202865 IC50 = 520 nM T37693 C02GKP 11203203 Ki > 1000 nM T37693 C73YFI 11213299 Ki = 326 nM T37693 CEPJ47 11224779 Ki = 242 nM T37693 CQ4KW2 11235490 EC50 = 158.49 nM T37693 C2AXJ6 11236772 Ki > 1000 nM T37693 CI8YG6 11237129 Ki > 1000 nM T37693 CYE8Q0 11244542 Ki = 5430 nM T37693 C0UM9Z 11246347 Ki = 26.9 nM T37693 C8IQ7N 11247557 EC50 = 251.19 nM T37693 C58AUX 11247638 Ki > 10000 nM T37693 C7VTE6 11247889 Ki = 240 nM T37693 C5KOE4 11249677 Ki = 1984 nM T37693 CRI87L 11259422 EC50 = 158.49 nM T37693 CC4Q6B 11260007 IC50 = 1100 nM T37693 CGB7Y1 11268746 Ki = 7.194 nM T37693 C2B6EC 11271934 Ki = 634 nM T37693 C9VEK5 11272442 Ki = 5444 nM T37693 CUH21X 11280135 Ki = 0.4898 nM T37693 CEJ4I7 11283445 IC50 = 1400 nM T37693 CWL54N 11293531 Ki = 815 nM T37693 CIA60C 11293559 Ki > 10000 nM T37693 CC2J3W 11294205 Ki = 608 nM T37693 C8E9AG 11294616 Ki = 906 nM T37693 CZY4N1 11294721 Ki > 1000 nM T37693 CBE45P 11295405 Ki = 3562 nM T37693 C1T9CA 11305400 Ki = 765 nM T37693 C6J3MW 11306088 Ki = 349 nM T37693 C8FS1B 11306174 Ki > 1000 nM T37693 CZX1D7 11313905 Ki = 138.04 nM T37693 C4H5FT 11318758 IC50 = 3200 nM T37693 CVH2C4 11321422 Ki >= 10000 nM T37693 CKUA15 11327582 EC50 = 199.53 nM T37693 C9NW2C 11329073 Ki = 3469 nM T37693 CN6G7L 11329858 Ki > 1000 nM T37693 CT8G0R 11338511 Ki = 4150 nM T37693 CTQE86 11340501 Ki = 230 nM T37693 C4J9LE 11341568 IC50 = 3600 nM T37693 C4G2KL 11349671 EC50 = 158.49 nM T37693 CA65US 11362251 Ki = 0.7499 nM T37693 C8AT6N 11363773 Ki > 1000 nM T37693 CE5VR2 11372171 Ki = 1.901 nM T37693 C25BJV 11373824 Ki = 0.08492 nM T37693 CQ26XK 11374417 Ki > 10000 nM T37693 C2SZV5 11375130 Ki = 823 nM T37693 CFA54H 11375615 Ki = 489 nM T37693 C7I9QK 11384486 Ki > 10000 nM T37693 C8AZP3 11386027 Ki = 505 nM T37693 CB1T7I 11386417 Ki = 696 nM T37693 C7ZY4I 11386749 IC50 = 5400 nM T37693 CB26AX 11391631 Ki > 10000 nM T37693 C37COB 11407971 Ki > 10000 nM T37693 CD49YO 11408036 Ki > 10000 nM T37693 CBN67Q 11408950 Ki = 430 nM T37693 CO6Z0Q 11409827 Ki > 1000 nM T37693 CE7B0I 11410344 IC50 = 6200 nM T37693 CY2ZI0 11413953 Ki = 57 nM T37693 CUSQ84 11430331 EC50 = 199.53 nM T37693 C35TRL 11443469 IC50 = 1100 nM T37693 CUN08B 11444148 IC50 = 1500 nM T37693 CU2P3D 11451762 Ki = 14 nM T37693 CQUG13 11454267 IC50 = 380 nM T37693 CP3V7Z 11464072 Ki = 2.399 nM T37693 C28OZA 11464704 Ki > 10000 nM T37693 C4R5FJ 11467430 IC50 = 5100 nM T37693 C6P2ZU 11473309 Ki = 16 nM T37693 CFT60D 11475997 Ki = 1650 nM T37693 C61OKL 11476787 Ki = 208 nM T37693 CGC2Z6 11477574 IC50 = 1400 nM T37693 CO8H9L 11488131 Ki > 10000 nM T37693 C9D2PH 11488705 IC50 = 44 nM T37693 C0VYA5 11493699 Ki = 960 nM T37693 CQO3I6 11493987 Ki = 19.5 nM T37693 CH0R5A 11494137 Ki = 3.162 nM T37693 CAR63Q 11494221 IC50 = 26 nM T37693 CN86KZ 11494391 Ki > 1000 nM T37693 CRLQ46 11494777 IC50 = 9000 nM T37693 CH79ND 11495004 Ki = 295.12 nM T37693 C2K5TP 11495157 Ki = 426 nM T37693 C5B6XG 11495398 Ki = 30 nM T37693 C0C2AR 11495877 IC50 = 69 nM T37693 CJ1OG8 11496202 Ki = 6600 nM T37693 CN3K8T 11496328 Ki = 5372 nM T37693 CBD28Z 11496638 Ki = 3526 nM T37693 CCQ85R 11501072 Ki = 0.3981 nM T37693 CTYJ07 11501580 EC50 = 5 nM T37693 CH21BN 11501747 EC50 = 3.1 nM T37693 C9Q0WB 11502034 Ki = 14 nM T37693 C1Z9YC 11502689 Ki = 420 nM T37693 C9X2RT 11503256 IC50 = 25.12 nM T37693 C0ZKG3 11504660 EC50 = 19540 nM T37693 CNM0C3 11507880 Ki = 218.78 nM T37693 CV8I4Q 11507883 Ki = 1.9 nM T37693 CCDQ14 11508636 Ki = 2.754 nM T37693 C47RUL 11508949 Ki = 0.51 nM T37693 C7Y9AS 11509456 IC50 = 12.59 nM T37693 C1TC7Y 11510814 EC50 = 20920 nM T37693 CJ48YV 11515193 Ki > 10000 nM T37693 C1SF2Q 11515395 Ki = 0.7079 nM T37693 C4U2YJ 11515910 Ki = 0.18 nM T37693 CDT27M 11516830 Ki = 238 nM T37693 C6D2HV 11517770 IC50 = 19.95 nM T37693 CB03ES 11517940 Ki = 9.3 nM T37693 C23UNF 11517964 Ki = 6.3 nM T37693 CXI1O0 11522517 Ki = 1.3 nM T37693 C2YZM1 11522943 Ki = 0.99 nM T37693 CMEY72 11523234 Ki = 11 nM T37693 CATI07 11524428 Ki = 584 nM T37693 C20FDW 11524622 Ki = 2700 nM T37693 CAJO54 11525340 Ki = 10000 nM T37693 CA7LK1 11529923 Ki = 0.14 nM T37693 C8QL3R 11530348 Ki = 3570 nM T37693 CR0E5G 11530365 Ki > 1000 nM T37693 CYR8X5 11530502 Ki = 1.9 nM T37693 CAN23D 11532254 IC50 = 65 nM T37693 CQ8L3J 11532557 Ki = 430 nM T37693 C2UF3G 11533229 Ki = 2490 nM T37693 CK53RQ 11537652 Ki = 0.4786 nM T37693 CVTA54 11537904 Ki = 25.7 nM T37693 C2C7YA 11541635 Ki = 1.7 nM T37693 CSH2A1 11544639 Ki = 0.21 nM T37693 CU49XP 11545113 Ki = 181 nM T37693 CD1QL5 11546775 Ki = 3.02 nM T37693 CB1DF3 11551160 Ki = 3.1 nM T37693 CTS15V 11551962 Ki = 30.9 nM T37693 CNHP10 11552423 Ki = 32 nM T37693 C7V3EQ 11553430 Ki = 11.2 nM T37693 CQW9O7 11553971 Ki = 67 nM T37693 C6GF0S 11559386 Ki = 0.08511 nM T37693 CCB6F1 11559434 Ki = 0.1479 nM T37693 CV06DX 11559474 Ki = 8.3 nM T37693 CVX3N5 11559687 Ki > 1000 nM T37693 C7ZIX8 11559736 Ki = 455 nM T37693 CT0YQ3 11560122 IC50 > 8900 nM T37693 C31FJV 11560244 Ki = 4.7 nM T37693 CON1Q8 11560246 Ki = 13.4 nM T37693 CYUF67 11560249 Ki > 10000 nM T37693 C2XCT3 11560942 IC50 = 3981.07 nM T37693 C3XD0O 11573397 Ki = 3.8 nM T37693 CJ59DW 11574104 Ki = 201 nM T37693 C5Y2NL 11574170 EC50 = 77 nM T37693 CS2T3B 11574895 Ki = 6 nM T37693 CGF9C0 11575063 Ki = 160 nM T37693 C9JS7A 11576961 Ki > 1000 nM T37693 C3VA1R 11580465 EC50 = 2.1 nM T37693 CV8G3F 11580822 EC50 = 2.9 nM T37693 CBS81K 11581197 Ki = 3.89 nM T37693 CV0A1L 11581982 IC50 = 63.1 nM T37693 CCM0H1 11582155 Ki = 400 nM T37693 CBF4O5 11583616 EC50 = 23670 nM T37693 CK95VZ 11583984 Ki = 17.9 nM T37693 C8XGZ6 11585047 Ki = 0.4 nM T37693 C3M6LW 11588379 Ki = 53.7 nM T37693 C1H8NL 11589048 Ki = 46.77 nM T37693 C4WHZ5 11591162 IC50 = 2156.1 nM T37693 C4EA7K 11595816 Ki = 0.1 nM T37693 CWV6T3 11595817 Ki = 3.3 nM T37693 CO6B1E 11595958 Ki > 1000 nM T37693 C0HFJ8 11597339 Ki = 340 nM T37693 CF8L2I 11597475 Ki = 1.259 nM T37693 CU37FZ 11597700 Ki = 1400 nM T37693 C4CN3F 11601669 Ki = 574 nM T37693 CU4I5W 11602703 Ki = 102.33 nM T37693 C0R1NH 11603123 Ki = 4.571 nM T37693 C4TN2S 11603482 IC50 = 260 nM T37693 CXL1Q2 11604689 EC50 = 2.5 nM T37693 C62OPJ 11609691 Ki = 1.778 nM T37693 C3FZJ9 11610001 Ki = 1.778 nM T37693 CMZ06K 11610023 Ki = 2.239 nM T37693 CN5U8O 11610189 IC50 = 82 nM T37693 CY8F1N 11611314 Ki > 1000 nM T37693 CGZ98H 11611505 IC50 = 1800 nM T37693 CSGU46 11612182 IC50 = 100 nM T37693 CRF2D3 11612574 Ki = 1032 nM T37693 CV4K9F 11616911 Ki = 8.128 nM T37693 CW1M9F 11617449 IC50 = 38 nM T37693 CESR67 11617925 Ki = 0.9 nM T37693 C8J9QA 11618679 IC50 = 0.7943 nM T37693 CH0I6J 11620691 IC50 = 704.9 nM T37693 C23WZM 11625937 Ki = 3.9 nM T37693 C93NWK 11626344 IC50 = 398.11 nM T37693 C14MPD 11626933 Ki = 2110 nM T37693 COF90W 11631918 Ki = 784 nM T37693 C8R1OK 11632670 Ki = 1.38 nM T37693 CMZ42U 11632980 Ki = 125 nM T37693 CA7K6Y 11638547 Ki = 5400 nM T37693 CX1K2J 11639250 Ki = 26.92 nM T37693 C5K9JX 11641397 Ki > 1000 nM T37693 CP1X4A 11646462 Ki = 2.5 nM T37693 C8Q0BW 11648843 Ki = 72 nM T37693 C2IJK0 11653150 Ki = 540 nM T37693 CNOU53 11653233 Ki = 3.86 nM T37693 CYD30X 11653936 IC50 = 110 nM T37693 C52VFG 11654304 Ki = 13 nM T37693 C1Q3HS 11655065 IC50 = 340 nM T37693 CWNX26 11659823 Ki = 51 nM T37693 C7ZI9D 11660288 EC50 = 3.2 nM T37693 CF59VR 11660635 Ki = 18 nM T37693 C7N8JK 11660978 Ki = 371 nM T37693 C83IZM 11661005 Ki > 10000 nM T37693 CD8EV7 11666821 Ki > 10000 nM T37693 CJW09U 11667488 Ki = 6430 nM T37693 CIX9F1 11667698 EC50 = 0.2512 nM T37693 CYR0S8 11668868 Ki = 350 nM T37693 CE7J1F 11669478 Ki = 0.88 nM T37693 CV01BZ 11670102 Ki = 182 nM T37693 C59LNI 11673821 Ki = 2.1 nM T37693 C5TO0E 11674728 Ki > 10000 nM T37693 CP5SQ2 11675463 Ki = 41.7 nM T37693 CM4OQ3 11675994 Ki = 0.87 nM T37693 C0NOQ3 11676975 Ki = 2.9 nM T37693 C1YVP6 11677439 EC50 = 25930 nM T37693 CO0Z4M 11683132 Ki = 100 nM T37693 CYJ2U8 11683348 Ki = 260 nM T37693 CEJ3R7 11683612 IC50 = 330 nM T37693 CLB8K0 11688907 Ki = 2.754 nM T37693 CG8ZF9 11689178 Ki > 1000 nM T37693 C3WBU8 11689242 EC50 = 11 nM T37693 CBW6K3 11689539 Ki = 1.585 nM T37693 CJ70LG 11689920 Ki > 1000 nM T37693 C76LTP 11690128 Ki > 5000 nM T37693 CYB9E3 11692359 Ki = 11 nM T37693 C4CBE3 11695365 Ki > 10000 nM T37693 CSNO87 11696383 Ki = 109 nM T37693 CMA60S 11696747 IC50 = 1400 nM T37693 CZS68I 11697361 Ki = 0.3 nM T37693 C15KDM 11697527 Ki = 0.4797 nM T37693 CXRS16 11703427 Ki = 9.333 nM T37693 CX3J6Z 11703995 Ki = 844 nM T37693 C53ZLN 11705255 Ki = 1321 nM T37693 CHO5Q9 11705479 Ki > 10000 nM T37693 CK7Z6O 11706218 EC50 = 23210 nM T37693 CGI8A7 11708992 Ki = 56 nM T37693 C9Y7AC 11710203 Ki = 772 nM T37693 CO40LS 11710271 EC50 = 16.8 nM T37693 CJE5D9 11712296 Ki = 1086 nM T37693 CQZ7T6 11716831 Ki = 3.3 nM T37693 CWRB76 11718456 IC50 = 0.631 nM T37693 CY7KA2 11719546 Ki = 3495 nM T37693 CE2H4Y 11719679 Ki = 200 nM T37693 CV71DR 11725464 Ki = 5.5 nM T37693 C4H1UG 11729245 Ki = 3110 nM T37693 CSA9Z2 11729545 Ki = 6061 nM T37693 C7C4PI 11732080 Ki > 5000 nM T37693 CSRB59 11743928 Ki = 12 nM T37693 C3L6FB 11748721 Ki = 2570 nM T37693 C6AXN2 11756059 IC50 = 3300 nM T37693 CLM20Y 11756106 Ki = 0.5 nM T37693 CQ41EZ 11756763 Ki = 13 nM T37693 C7VIS9 11762170 Ki = 2190 nM T37693 C7L0UM 11784543 Ki = 3959 nM T37693 C8K4IE 11785274 IC50 = 720 nM T37693 CP30IU 11785628 IC50 = 2500 nM T37693 C9P6WX 11825838 Ki > 5000 nM T37693 C2FVO0 11830207 Ki > 10000 nM T37693 CO7P6C 11842620 Ki > 10000 nM T37693 CL6Z1P 11949889 Ki > 10000 nM T37693 CNW8M4 11950060 Ki > 10000 nM T37693 C9EN7I 11950589 Ki > 10000 nM T37693 CF7I2Q 11950590 Ki > 10000 nM T37693 C89NBK 11950958 IC50 = 2390 nM T37693 C0RNE1 11951124 Ki > 7000 nM T37693 CM0YF9 11951128 Ki = 2080 nM T37693 CBV53O 11951300 Ki > 5000 nM T37693 CGHC56 11951302 Ki > 10000 nM T37693 C74VTU 11951655 Ki > 10000 nM T37693 C1MTD0 11951656 Ki > 10000 nM T37693 CFNY34 11951657 Ki > 10000 nM T37693 C0DEG8 11951661 Ki > 10000 nM T37693 CHVG30 11952383 Ki > 7000 nM T37693 CN2S4P 11982685 Ki = 780 nM T37693 CD6Y4G 11995766 IC50 = 1410 nM T37693 C0FMG3 11996213 EC50 = 0.7943 nM T37693 C68UFD 11996214 Ki = 20 nM T37693 CY5VJ7 11996215 EC50 = 6.31 nM T37693 C3U2ZK 11996349 Ki = 23.8 nM T37693 CDBZ94 11996350 Ki = 8.4 nM T37693 CJO56E 11996351 EC50 = 0.1995 nM T37693 C5KR9H 12000834 Ki = 20600 nM T37693 CHC8O9 12000836 Ki = 5400 nM T37693 C6RO3B 12000837 Ki = 16600 nM T37693 CAQH93 12000925 Ki = 75600 nM T37693 C53JEN 12000927 Ki > 30000 nM T37693 CGN62B 12001013 Ki = 14700 nM T37693 C7S9TZ 12146779 Ki = 4880 nM T37693 C2R4EN 12146780 Ki = 2090 nM T37693 CLHV82 12146781 IC50 = 322 nM T37693 C5P2CA 12146782 Ki = 48 nM T37693 C5IL3V 12146783 IC50 = 6.1 nM T37693 C5FWA0 12216569 Ki = 12670 nM T37693 CKG9Q1 12232068 Ki >= 10000 nM T37693 C1B3EX 12315250 Ki = 4535 nM T37693 CRO26B 12471990 Ki > 10000 nM T37693 C2CQS6 12495545 EC50 = 3981.07 nM T37693 CEZD35 12971995 EC50 = 14 nM T37693 C5RJ6P 13045465 Ki > 10000 nM T37693 C9CAK4 13166820 Ki >= 10000 nM T37693 CPD42A 13188551 Ki = 132.2 nM T37693 C8V5UW 13611813 Ki = 9929.99 nM T37693 C2WB4I 13713752 Ki > 5000 nM T37693 C9MQO2 14135316 IC50 = 224 nM T37693 CF3W4S 14135317 IC50 = 197 nM T37693 C2TY8N 14135320 IC50 = 9100 nM T37693 CI0LC3 14378151 Ki = 7.4 nM T37693 CC5Q7O 14417955 Ki >= 10000 nM T37693 C0XNF5 14417956 Ki > 10000 nM T37693 CKP12X 14589394 Ki = 158 nM T37693 CF1EO5 14852550 Ki > 10000 nM T37693 C9C0DT 14898643 Ki > 10000 nM T37693 C5RCD3 14898644 Ki > 10000 nM T37693 C7Q8HG 14950683 Ki > 10000 nM T37693 CG49IS 14950684 Ki > 10000 nM T37693 CLK42M 14950685 Ki > 10000 nM T37693 CD13NW 14950686 Ki = 16600 nM T37693 C5THR8 15000083 Ki = 2.61 nM T37693 CP86TW 15000084 Ki = 51 nM T37693 C39MRN 15262805 Ki > 10000 nM T37693 CB0I3R 15341903 Ki = 69 nM T37693 CIEM61 15481172 Ki = 1090.5 nM T37693 CV25BT 15603837 Ki > 10000 nM T37693 C1QR0W 15614389 EC50 = 0.078 nM T37693 CGHE06 15953828 EC50 = 10 nM T37693 C6NL8T 15991674 Ki = 6600 nM T37693 CWP5Q0 15991676 Ki = 19100 nM T37693 C20ZAI 15998061 Ki = 9900 nM T37693 CX2CF4 15998383 Ki = 22800 nM T37693 C0PU4I 15998702 Ki = 7400 nM T37693 CP1X7K 16000037 Ki = 10000 nM T37693 CC6O9T 16045226 Ki = 19.95 nM T37693 CJ78MO 16045297 Ki = 6.31 nM T37693 C02YSU 16046254 EC50 = 6.6 nM T37693 CIJM09 16067243 Ki > 10000 nM T37693 CV2QE8 16067244 Ki > 10000 nM T37693 CTX4V2 16067267 Ki = 1030 nM T37693 CPLV09 16067270 Ki = 5810 nM T37693 CM9XK7 16067272 Ki > 10000 nM T37693 CZ7E3U 16067273 Ki > 10000 nM T37693 CF4JZ3 16089262 Ki = 1800 nM T37693 CI9O5Y 16089263 Ki = 14900 nM T37693 C9Y4WC 16094766 Ki = 131825673.9 nM T37693 C1R4QA 16098312 IC50 > 2000 nM T37693 CCU10Q 16098313 IC50 = 600 nM T37693 C8JMW2 16098324 IC50 = 770 nM T37693 COK4S9 16098325 IC50 = 1700 nM T37693 CJ27GS 16098334 IC50 = 190 nM T37693 C0U3AZ 16098336 IC50 = 290 nM T37693 CM1PN6 16098337 IC50 = 88 nM T37693 C65WRB 16098343 IC50 = 100 nM T37693 CTHC39 16098344 IC50 = 140 nM T37693 CTZ95W 16098380 IC50 = 450 nM T37693 C4H5XE 16098381 IC50 = 200 nM T37693 CHW52V 16114441 EC50 < 1000 nM T37693 CRI63Z 16126849 EC50 = 330 nM T37693 CMH38I 16367681 Ki > 10000 nM T37693 C9APD3 16482860 IC50 > 10000 nM T37693 C3GN7A 16644329 Ki > 10000 nM T37693 CLY6K7 16659101 Ki = 1300 nM T37693 CQG04A 16719315 EC50 = 630 nM T37693 CP24ZG 16719316 EC50 = 400 nM T37693 C4D1JF 16719551 EC50 > 25000 nM T37693 C2GH8E 16719552 EC50 = 400 nM T37693 C6GD8W 16719553 EC50 > 25000 nM T37693 CAPU50 16719554 EC50 = 125 nM T37693 CN95DG 16719649 EC50 = 200 nM T37693 C4YS1C 16720930 EC50 > 25000 nM T37693 CSG68P 16720931 EC50 > 25000 nM T37693 C9HB5D 16720932 EC50 = 5000 nM T37693 C34UKV 16720933 EC50 = 80 nM T37693 CQ7G9D 16720934 EC50 = 400 nM T37693 CNVB32 16720935 EC50 = 400 nM T37693 C8EK4I 16725534 EC50 = 29440 nM T37693 C2F5LA 16737690 IC50 > 10000 nM T37693 CHU72I 16738321 IC50 = 470 nM T37693 CY32BQ 16738395 IC50 > 10000 nM T37693 CGC6A8 16739312 IC50 = 394.4 nM T37693 CTF3J5 16752693 EC50 = 4 nM T37693 CK8M6J 16866369 EC50 = 86 nM T37693 CEO7I5 17352616 EC50 > 10000 nM T37693 CYA04E 17386953 Ki = 3081 nM T37693 C28ZHR 17450266 Ki = 120 nM T37693 C6JFW2 17592519 Ki > 10000 nM T37693 C9UGI2 17754357 Ki = 0.64 nM T37693 CEL3S7 17757539 Ki = 2400 nM T37693 C8WBK9 17984783 EC50 = 100 nM T37693 CD9T6M 17984800 EC50 = 50.12 nM T37693 CY7RP4 18407247 Ki > 1000 nM T37693 C51JGA 18839400 Ki = 313 nM T37693 CMU2Z1 19363234 Ki = 0.1099 nM T37693 CA97PZ 19363251 Ki = 0.4395 nM T37693 C47RWC 19363289 Ki = 2.5 nM T37693 C0A6DC 19363292 Ki = 14 nM T37693 C3BD1L 19363351 Ki = 8.395 nM T37693 CZ2PL8 19363367 Ki = 1.799 nM T37693 C6JCP8 19363402 Ki = 0.0879 nM T37693 CRXU83 19363412 Ki = 4.797 nM T37693 C18BYE 19363420 Ki = 7.295 nM T37693 C9MQ6T 19363480 Ki = 10.99 nM T37693 CTV3G1 19363528 Ki = 3.698 nM T37693 CD89PR 19438815 Ki = 22 nM T37693 C4H3AL 19868648 Ki = 6.8 nM T37693 CJ2IL9 20386375 Ki > 3000 nM T37693 C0GHP8 20442464 EC50 = 6309.57 nM T37693 CI17MH 21035228 Ki = 179 nM T37693 C0YC6G 21815908 Ki = 420 nM T37693 CTL0C7 21858022 Ki > 10000 nM T37693 CF2S3C 21858023 Ki > 10000 nM T37693 C3YPZ2 21868807 Ki > 10000 nM T37693 C8BW6H 21948996 Ki = 7504 nM T37693 C94KPY 21949023 Ki = 1412 nM T37693 C6N2GY 21949029 Ki = 1072 nM T37693 C1OW2Z 21949050 Ki = 1811 nM T37693 CJAZ80 21949054 Ki = 54 nM T37693 C45PAW 21984801 IC50 = 1300 nM T37693 CZFS96 21984889 IC50 = 5100 nM T37693 CJ6HK9 22038546 Ki = 850 nM T37693 CMW59D 22181270 EC50 = 24 nM T37693 CFI69E 22181275 EC50 = 6.2 nM T37693 C0QOK7 22181282 Ki = 57 nM T37693 CL52WO 22181288 Ki = 4342 nM T37693 C84HYE 22181294 EC50 = 3.3 nM T37693 CL45HJ 22181304 EC50 = 2.9 nM T37693 C8OGN3 22181310 EC50 = 25 nM T37693 CSW3J7 22181316 Ki > 5000 nM T37693 CQRK86 22181322 EC50 = 25 nM T37693 CGC04B 22181344 EC50 = 5 nM T37693 C19BHA 22181345 EC50 = 52 nM T37693 C4S5NI 22181387 EC50 = 4.2 nM T37693 CX68DC 22181394 Ki = 36 nM T37693 C9FX1Q 22181403 Ki = 5.7 nM T37693 CX1U8F 22181408 EC50 = 18 nM T37693 CO87EI 22181435 EC50 = 2.1 nM T37693 CYUW32 22181436 Ki = 188 nM T37693 C9D4OS 22266461 Ki = 235 nM T37693 CQR90C 22266472 Ki = 976 nM T37693 CU61ZM 22266537 Ki = 40 nM T37693 CPT56H 22266539 Ki = 236 nM T37693 C7K3PT 22267343 Ki = 3270 nM T37693 C6WLG2 22267384 Ki = 1601 nM T37693 CUV02J 22267389 Ki = 2755 nM T37693 CLI1M8 22267402 Ki = 3835 nM T37693 C78LFV 22267403 Ki = 2864 nM T37693 CIH20L 22285476 Ki = 1100 nM T37693 C9O5TA 22422463 Ki = 6000 nM T37693 C26KER 22422464 Ki = 4800 nM T37693 C64NHO 22422466 Ki = 4000 nM T37693 C1U4XQ 22431127 EC50 = 110 nM T37693 C27SAH 22474540 EC50 = 0.77 nM T37693 CX38ZN 22848569 Ki > 10000 nM T37693 CV2E0N 22969459 EC50 = 8 nM T37693 CK92XJ 23231044 Ki > 1000 nM T37693 C1ZT0J 23231127 Ki > 1000 nM T37693 C0RL6E 23281241 Ki > 1000 nM T37693 CJO3Z6 23328304 Ki = 1000 nM T37693 C5OWG2 23398409 Ki = 5100 nM T37693 C9H8QR 23398410 Ki = 1200 nM T37693 CU8I1Z 23398439 Ki = 2300 nM T37693 C26JDS 23555588 Ki = 0.02 nM T37693 CEHV12 23555590 Ki = 0.1799 nM T37693 CXDB37 23555594 Ki = 5 nM T37693 C1VTH7 23555596 Ki = 0.02099 nM T37693 CVB8K1 23555598 Ki = 0.021 nM T37693 C74MCD 23555607 Ki = 0.2198 nM T37693 CA69IO 23585153 EC50 = 30 nM T37693 CA1F0L 23585155 EC50 = 6 nM T37693 CQLO71 23585201 EC50 = 3 nM T37693 C3Z5CX 23585203 EC50 = 3 nM T37693 CCH5I9 23585204 EC50 = 25 nM T37693 COB53R 23587763 Ki = 0.2 nM T37693 C2MC4Q 23588031 Ki = 20 nM T37693 C82JLB 23620581 Ki = 3219 nM T37693 CX8MY0 23626079 Ki = 270 nM T37693 C8IVH5 23628267 Ki = 0.81 nM T37693 CXDT91 23634661 Ki = 966 nM T37693 CBG3F0 23634663 Ki > 2000 nM T37693 CL5SW0 23634664 Ki = 1670 nM T37693 C7QC4Z 23634776 Ki > 2000 nM T37693 CY7B8I 23634782 Ki < 2000 nM T37693 CI6TE1 23634784 Ki = 152 nM T37693 CFKT02 23634786 Ki > 4000 nM T37693 CZS87H 23634906 Ki = 144 nM T37693 C3M9DF 23635640 Ki = 21.6 nM T37693 C1LQJ3 23635769 Ki = 14 nM T37693 CN2LR8 23635897 Ki = 663 nM T37693 CP2O9Z 23635898 Ki > 2000 nM T37693 CM8SE1 23635899 Ki > 3000 nM T37693 CJ32OK 23635900 Ki = 338 nM T37693 CNU60E 23636025 Ki = 25.5 nM T37693 C1U8HS 23636026 Ki = 1130 nM T37693 CB4L8Z 23636027 Ki = 265 nM T37693 CW0JB8 23636029 Ki = 1670 nM T37693 C89APR 23636259 Ki = 26.1 nM T37693 C2O4RT 23636260 Ki = 121 nM T37693 C93XVD 23636504 Ki = 1550 nM T37693 CQG41O 23636505 Ki = 582 nM T37693 CS0W5U 23636506 Ki = 656 nM T37693 C8WGQ1 23636507 Ki = 225 nM T37693 CR0BT2 23636508 Ki = 1120 nM T37693 CN8F6O 23642627 Ki = 27.4 nM T37693 CGN80J 23643046 Ki = 4760 nM T37693 CJ0QV7 23654188 Ki > 1000 nM T37693 CMC87P 23654862 Ki = 634 nM T37693 C1LVE4 23656391 Ki = 6 nM T37693 CA0VJ4 23730229 Ki = 21700 nM T37693 CTKS21 23848377 Ki = 320 nM T37693 CY48RZ 23968873 Ki > 10000 nM T37693 C52FSE 24096428 Ki = 0.4898 nM T37693 CBU1K9 24125805 EC50 = 436.5 nM T37693 C0DN4V 24180486 EC50 = 7.2 nM T37693 C9G3DP 24400240 EC50 = 6 nM T37693 C2CV7N 24467372 Ki > 10000 nM T37693 C8P4FA 24531721 Ki > 1000 nM T37693 CIP5B0 24748172 Ki > 1000 nM T37693 C42DBF 24748217 EC50 = 6.31 nM T37693 C2FG6X 24750597 EC50 = 0.91 nM T37693 CVNT09 24763642 EC50 = 1.8 nM T37693 CT4SJ0 24766011 Ki = 422 nM T37693 CFN89K 24768454 Ki > 3940 nM T37693 CNC6R4 24768455 Ki > 3940 nM T37693 CUE3X8 24768456 Ki > 3940 nM T37693 C5W8OH 24768457 Ki = 3940 nM T37693 C7XE2U 24768458 Ki > 3940 nM T37693 CGF2B5 24768459 Ki = 1750 nM T37693 CVD3X5 24768460 Ki = 2180 nM T37693 CW35HD 24768461 Ki = 390 nM T37693 CC28YT 24768462 Ki > 3940 nM T37693 CU5P9T 24768463 Ki > 3940 nM T37693 CY3CP1 24768464 Ki > 3940 nM T37693 C8G6CH 24768465 IC50 = 200 nM T37693 CBU2P6 24768466 Ki = 510 nM T37693 C80IVA 24768467 Ki = 64 nM T37693 CFN6B5 24768468 Ki = 980 nM T37693 C5S0WL 24768469 Ki = 3940 nM T37693 C61ELO 24768470 Ki = 87 nM T37693 CS6UN4 24768471 Ki = 20 nM T37693 CX79AV 24768472 Ki = 150 nM T37693 CSM3C5 24768473 Ki = 1.7 nM T37693 CR63JT 24768474 Ki = 29 nM T37693 C4CKN2 24768475 Ki = 1370 nM T37693 CGZ9X6 24768476 Ki = 1.3 nM T37693 C8I4XR 24768477 Ki = 2400 nM T37693 C4K6QC 24768478 Ki > 3940 nM T37693 C09CZR 24768479 Ki = 390 nM T37693 C1PR3H 24768480 Ki = 65 nM T37693 C69VXF 24768481 Ki = 3940 nM T37693 CPBI12 24768482 Ki = 3940 nM T37693 CWO6X4 24768483 Ki = 570 nM T37693 C6GKY8 24768484 Ki > 3940 nM T37693 C8IS0O 24768485 Ki > 3940 nM T37693 CVIH02 24768486 Ki = 3940 nM T37693 CV6HK2 24768487 Ki = 390 nM T37693 CC1B9L 24768488 Ki = 4.898 nM T37693 CHQ5E7 24768489 Ki = 1.585 nM T37693 CS94WN 24768490 Ki = 3 nM T37693 CX86RC 24768491 Ki = 6.6 nM T37693 CR1N5H 24768492 Ki = 0.6457 nM T37693 CGJ93M 24768493 Ki = 3.467 nM T37693 C95JFQ 24768494 Ki = 2.951 nM T37693 CBA0J3 24768495 Ki = 1.778 nM T37693 CIC1H5 24768496 Ki = 0.6918 nM T37693 CZAT71 24768497 Ki = 21 nM T37693 C3UIX7 24768498 Ki = 1 nM T37693 CVGO46 24768499 Ki = 9 nM T37693 CX5N8F 24768500 Ki = 91.2 nM T37693 C4E0SL 24768501 Ki = 234.42 nM T37693 CX9CH8 24768502 Ki > 1000 nM T37693 C6AR0N 24768503 Ki > 1000 nM T37693 C4U9RH 24768504 Ki < 1000 nM T37693 C6X8BW 24768505 Ki = 30 nM T37693 C8DJL5 24768506 Ki < 1000 nM T37693 CT6OR5 24768507 EC50 = 73 nM T37693 C1I4VG 24768508 Ki = 25 nM T37693 CXAD71 24768509 Ki = 58 nM T37693 CQLB52 24768510 Ki = 5 nM T37693 CRIJ68 24768511 Ki = 61.66 nM T37693 CCV3R8 24768512 Ki = 0.4 nM T37693 C8WTX4 24771838 EC50 = 65 nM T37693 C6NQZ2 24779702 EC50 = 0.5 nM T37693 CGLZ78 24779731 EC50 = 10 nM T37693 C02APD 24794709 EC50 = 0.3 nM T37693 C4V0AG 24794743 EC50 = 1.3 nM T37693 CI3SF5 24797443 Ki > 10000 nM T37693 C52FXR 24801854 EC50 = 135 nM T37693 CY93EF 24809843 Ki = 21.48 nM T37693 C41PZC 24810237 IC50 = 818 nM T37693 C2V5HT 24810792 IC50 > 10000 nM T37693 C2NQ6G 24825767 Ki > 1000 nM T37693 C52OSW 24828563 Ki > 3 nM T37693 CH9P2T 24849046 Ki > 10000 nM T37693 CIC0B1 24856117 EC50 = 11 nM T37693 C60CQO 24856504 Ki > 10000 nM T37693 CH1AO3 24856554 Ki > 10000 nM T37693 CZ7PQ6 24856591 Ki = 1260 nM T37693 C7WDN2 24856637 Ki > 10000 nM T37693 CM35KT 24856919 Ki > 10000 nM T37693 CQ7Z3J 24857160 Ki > 10000 nM T37693 CLN2Y9 24857341 Ki > 10000 nM T37693 C67SFU 24857887 EC50 = 2 nM T37693 CI9ZX3 24857902 Ki = 1900 nM T37693 C8XSM0 24857903 Ki = 4945 nM T37693 CR2LS5 24862715 Ki = 89 nM T37693 C4SR7K 24862938 IC50 = 4240 nM T37693 CLG5O2 24863156 Ki = 14.9 nM T37693 C3P4FQ 24863231 Ki = 6.3 nM T37693 CECW68 24863252 Ki = 3.54 nM T37693 C3IA4J 24863253 Ki = 0.88 nM T37693 CXA79O 24863254 Ki = 1.13 nM T37693 CTJ1M4 24863255 Ki = 1.68 nM T37693 CB0NW8 24863396 Ki = 74 nM T37693 CP4Z2L 24863434 EC50 = 0.7 nM T37693 C8UVA9 24863530 Ki = 260 nM T37693 CL2B6W 24863531 Ki = 53 nM T37693 CI2QU4 24863532 Ki = 36.6 nM T37693 C7Y2GK 24863613 Ki = 17.6 nM T37693 CMT60O 24863702 Ki = 35.6 nM T37693 CBI19Y 24863730 Ki = 371 nM T37693 C4QXJ2 24863966 Ki = 62 nM T37693 CFV5K0 24864017 Ki = 0.27 nM T37693 CBP1Y5 24865177 EC50 > 10000 nM T37693 CIY6F4 24865179 EC50 > 10000 nM T37693 C2D0YB 24873535 Ki = 11 nM T37693 CEM91N 24878075 EC50 = 215 nM T37693 CXV19G 24881409 Ki = 1044 nM T37693 CF5KN2 24881410 Ki = 1109 nM T37693 C1HA5X 24881411 Ki = 1124 nM T37693 CB4OX6 24881412 Ki = 1781 nM T37693 CX2QD9 24881413 Ki = 758 nM T37693 CJZ52T 24881469 Ki = 492 nM T37693 CV3QZ2 24884489 Ki = 24 nM T37693 C5OZ6A 24884501 Ki = 1.7 nM T37693 C4D8UX 24884502 Ki = 23 nM T37693 C25XLM 24890016 Ki > 10000 nM T37693 CZ50UW 24890182 Ki > 10000 nM T37693 C36SBO 24890183 Ki > 10000 nM T37693 CNQ6I4 24894028 Ki = 9 nM T37693 C3C0KP 24894134 EC50 = 7 nM T37693 CQY82F 24896430 Ki = 1.07 nM T37693 CJ8AB7 24901353 EC50 = 0.8 nM T37693 CK69LX 24944970 IC50 > 10000 nM T37693 CPT7H9 24944972 IC50 > 10000 nM T37693 CPL3Z0 24944973 IC50 > 10000 nM T37693 CR94OQ 24945940 EC50 = 60 nM T37693 CRD1G9 24946653 EC50 = 9.8 nM T37693 C7MU9F 24947740 EC50 = 136 nM T37693 C0UBF7 24947741 EC50 = 123 nM T37693 C65EYT 24947742 EC50 = 226 nM T37693 C85NPW 24952500 Ki = 7.9 nM T37693 CHPT23 24953766 Ki = 6 nM T37693 CM0NC1 24954444 EC50 = 140 nM T37693 C3SLV2 24954806 EC50 = 30 nM T37693 C8WH9Z 24954807 EC50 = 1600 nM T37693 CZ9EV5 24954808 EC50 = 10 nM T37693 COL0D1 24955167 EC50 = 200 nM T37693 C47VXF 24955168 EC50 = 50 nM T37693 CGF6L8 24955525 EC50 = 35 nM T37693 CW51DB 24955526 EC50 = 30 nM T37693 CJ36KQ 24955527 EC50 = 100 nM T37693 CR9Q8K 24955878 EC50 = 15000 nM T37693 C5RN6C 24956045 Ki = 1.9 nM T37693 C9AS5P 24956409 Ki = 67 nM T37693 CG9M3D 24956413 Ki = 1800 nM T37693 C4JC8Q 24965581 Ki = 1.2 nM T37693 CBW53M 24969357 IC50 = 9833 nM T37693 C8QV4P 24983869 IC50 = 5412.8 nM T37693 CPD69M 24984020 IC50 = 4234.4 nM T37693 CH56TG 24984021 IC50 = 901.7 nM T37693 CPTK86 24984022 IC50 = 1809.1 nM T37693 C3O5QS 24984023 IC50 = 1725.9 nM T37693 CO42TL 24984332 IC50 = 310.5 nM T37693 CR5MP8 24984333 IC50 = 919.6 nM T37693 CZ9DE6 24984334 IC50 = 1761.1 nM T37693 COQC35 24984485 IC50 = 1269.4 nM T37693 CS1OQ5 24984486 IC50 = 309.9 nM T37693 C7DSG8 24984487 IC50 = 385.9 nM T37693 C3BIU6 24990210 EC50 < 100 nM T37693 CZD3W7 24992427 IC50 = 2500 nM T37693 C9YMN0 24994351 IC50 = 3000 nM T37693 C2T0PY 24994664 IC50 = 8300 nM T37693 CY74AK 24994665 IC50 = 8000 nM T37693 C7VBJ3 24994981 IC50 = 3900 nM T37693 C5PUR9 24994982 IC50 = 4200 nM T37693 CZK8C0 24995602 IC50 = 4100 nM T37693 CUA84P 24995886 IC50 > 10000 nM T37693 C2LEI6 24995887 IC50 > 10000 nM T37693 CUMS01 24995912 IC50 = 2300 nM T37693 C62VTZ 24996234 IC50 = 1300 nM T37693 C2R6OP 24996235 IC50 = 4200 nM T37693 CU7I2A 24996238 IC50 = 3400 nM T37693 C34XJW 24996239 IC50 = 3300 nM T37693 C13YJI 24996565 IC50 = 7760 nM T37693 C7YU1S 25003672 EC50 = 0.04 nM T37693 CY9RK6 25003966 EC50 = 2284 nM T37693 CYP31X 25004304 EC50 = 5 nM T37693 C2DQP3 25004305 EC50 = 13 nM T37693 CC9R1L 25004638 EC50 = 1 nM T37693 CD6FI1 25004639 EC50 = 1.5 nM T37693 CER2X8 25004640 EC50 = 2 nM T37693 CP8L7C 25004979 EC50 = 14 nM T37693 CWOB35 25004981 EC50 = 0.4 nM T37693 C4EUD7 25005685 EC50 = 4 nM T37693 C6DVL4 25006674 Ki = 15.85 nM T37693 CETJ60 25006676 Ki = 50.12 nM T37693 CAB98T 25030040 Ki = 2.94 nM T37693 C9QM2T 25030041 Ki = 4.77 nM T37693 C40QGK 25033663 Ki = 52.6 nM T37693 CW1D6E 25033664 Ki = 0.8 nM T37693 CE14PW 25033665 Ki = 17.1 nM T37693 CBW5O1 25033667 Ki = 0.9 nM T37693 C1A0QO 25033736 Ki = 3.8 nM T37693 C3L4UA 25033812 EC50 = 270 nM T37693 C91HVB 25033813 EC50 = 2000 nM T37693 CBN0A5 25033871 EC50 > 10000 nM T37693 CG18DC 25033872 EC50 = 190 nM T37693 CP06NH 25033873 EC50 = 150 nM T37693 C6JAL1 25033874 EC50 = 670 nM T37693 C7G3DB 25033875 EC50 = 410 nM T37693 CJD73T 25033876 EC50 = 0.6 nM T37693 CTQ29P 25033938 EC50 = 0.33 nM T37693 CJ6S9L 25033939 EC50 = 2.4 nM T37693 C06YNQ 25033940 EC50 = 0.5 nM T37693 CZND73 25033941 EC50 = 3 nM T37693 CGX95B 25033942 EC50 = 10 nM T37693 C2N9UG 25033943 EC50 = 370 nM T37693 C2J1HF 25034003 EC50 = 78 nM T37693 CJ6G8M 25034004 EC50 = 14 nM T37693 CS9J8K 25034005 EC50 = 0.2 nM T37693 CBY1G8 25034006 EC50 = 31 nM T37693 C6RY5L 25034007 EC50 = 110 nM T37693 CJR0I9 25034070 EC50 = 11 nM T37693 CF7UY4 25034071 EC50 = 3.6 nM T37693 C2LB0M 25034073 EC50 > 10000 nM T37693 COCB26 25034074 EC50 = 470 nM T37693 CH09EK 25034075 EC50 = 200 nM T37693 CJF6E7 25034136 EC50 = 6 nM T37693 CY5RI2 25034137 EC50 = 4.8 nM T37693 CKBP28 25034138 EC50 = 0.089 nM T37693 COJC54 25034139 EC50 > 2.6 nM T37693 C0UG1V 25034140 EC50 = 0.6 nM T37693 CSF9M3 25034141 EC50 = 0.8 nM T37693 C7H3LM 25034205 EC50 = 38 nM T37693 CPO3V5 25034206 EC50 = 25 nM T37693 C3RZ9W 25034207 EC50 = 2.9 nM T37693 CHC78S 25034208 EC50 = 27 nM T37693 CCQ81R 25034209 EC50 = 1.7 nM T37693 CZ0JY9 25034273 EC50 = 4.9 nM T37693 CL45CE 25034494 Ki = 25.5 nM T37693 CX6RJ8 25034551 Ki = 6.3 nM T37693 CTZ5D6 25034552 Ki = 23.8 nM T37693 CI6RK0 25034553 Ki = 9.4 nM T37693 CN37RQ 25034554 Ki = 3.4 nM T37693 CY8C3F 25034555 Ki = 9.2 nM T37693 C7S6GR 25034601 Ki = 3.6 nM T37693 CA0M1S 25034602 Ki = 10.7 nM T37693 CH5CJ1 25034603 Ki = 24.2 nM T37693 C9FY7P 25034605 Ki = 1.6 nM T37693 CI9KQ0 25034658 Ki = 3.5 nM T37693 CVM70G 25034659 Ki = 55.9 nM T37693 CTOK52 25034660 Ki = 11.6 nM T37693 C8E4BW 25034661 Ki = 16.1 nM T37693 CW07TE 25034662 Ki = 14.3 nM T37693 CC14IN 25052853 IC50 = 2214 nM T37693 C1FU9T 25052854 IC50 = 1499.2 nM T37693 C8GU5B 25052855 IC50 = 6346 nM T37693 C3E8XA 25052856 IC50 = 3664.3 nM T37693 CHIM64 25052920 IC50 = 921 nM T37693 CF6GE2 25052921 IC50 = 1057.8 nM T37693 COL92Y 25052922 IC50 = 158 nM T37693 CGUL19 25052923 IC50 = 637.7 nM T37693 CF6AI2 25052924 IC50 = 278.3 nM T37693 C15YEA 25052990 IC50 = 1158.1 nM T37693 CM19FU 25052991 IC50 = 1576.4 nM T37693 CU28VO 25052992 IC50 = 1749.8 nM T37693 C01ADI 25052993 IC50 = 985.6 nM T37693 CS8C7R 25052995 IC50 = 2737.4 nM T37693 C8CSV3 25053066 IC50 = 7032.2 nM T37693 CQ36FL 25053067 IC50 = 785.1 nM T37693 C2YSM3 25053068 IC50 = 687.7 nM T37693 C1KZ0L 25053142 IC50 = 1206 nM T37693 CI8LQ6 25053143 IC50 = 4328.3 nM T37693 CX6F8W 25053144 IC50 = 564 nM T37693 CXFL75 25053145 IC50 = 260.6 nM T37693 CZ79SF 25053146 IC50 = 1900.1 nM T37693 C4WK5U 25053215 IC50 = 5719.5 nM T37693 CSB7F9 25053216 IC50 = 7179.1 nM T37693 C09NVD 25061041 IC50 = 4950 nM T37693 C7R6MK 25070947 EC50 = 9 nM T37693 CV4OA6 25094334 EC50 = 8.4 nM T37693 C30WTM 25094337 EC50 = 13 nM T37693 CY1FJ2 25094429 IC50 = 770 nM T37693 C6FZD5 25094431 IC50 = 891 nM T37693 C4UI7C 25094433 IC50 = 18000 nM T37693 C40JMD 25094607 EC50 = 2.4 nM T37693 CS2LZ4 25094611 EC50 = 2.9 nM T37693 C9ZTU4 25094701 IC50 = 9200 nM T37693 C5VIP4 25094884 EC50 = 1585 nM T37693 CTQB05 25095249 IC50 = 2400 nM T37693 CALF53 25095275 IC50 > 2000 nM T37693 CIK3S2 25095276 IC50 = 1800 nM T37693 C7MXU4 25095277 IC50 > 2000 nM T37693 CF2XN3 25095509 IC50 = 3400 nM T37693 CH0W1V 25095533 IC50 = 1800 nM T37693 CO76PH 25095792 IC50 = 2700 nM T37693 C3IF6X 25095795 IC50 > 2000 nM T37693 CBK9R7 25096563 IC50 = 9800 nM T37693 C9LUX8 25096565 IC50 = 8400 nM T37693 CRQ67O 25096567 IC50 = 6300 nM T37693 CDC4X6 25097842 IC50 = 4900 nM T37693 C1QX9B 25098113 IC50 > 2000 nM T37693 C51OER 25098115 IC50 > 2000 nM T37693 C2H6NK 25098369 IC50 = 5800 nM T37693 CE75CG 25098370 IC50 = 2700 nM T37693 C50QHA 25107503 Ki > 5000 nM T37693 C6ZWJ3 25107504 Ki > 5000 nM T37693 CMX36H 25107505 Ki > 5000 nM T37693 CHV9I0 25107506 Ki > 5000 nM T37693 C02LQB 25113749 IC50 > 10000 nM T37693 CG64CV 25132791 EC50 = 10 nM T37693 CMC96H 25135579 Ki = 828 nM T37693 CR9TP0 25136948 IC50 = 948 nM T37693 CS0Z2Y 25140206 Ki > 10000 nM T37693 CPB4N3 25140358 Ki > 10000 nM T37693 CDXE43 25140500 Ki > 10000 nM T37693 C3F4ZI 25140502 Ki = 7400 nM T37693 C9V1AJ 25141102 Ki = 0.71 nM T37693 C6K7FP 25141397 Ki = 3000 nM T37693 CXF18L 25149250 IC50 = 376 nM T37693 CQ6K0R 25149251 IC50 = 804 nM T37693 C7F8HT 25149339 IC50 = 680 nM T37693 CC9F0L 25149435 IC50 = 3320 nM T37693 C5D2JX 25149436 IC50 = 954 nM T37693 C7K2SW 25149437 IC50 = 1130 nM T37693 CHQ97G 25149438 IC50 = 1240 nM T37693 CRYN61 25149522 IC50 = 513 nM T37693 CHX64U 25149523 IC50 = 579 nM T37693 C08QES 25149524 IC50 = 1050 nM T37693 C6SY4U 25149821 IC50 = 1480 nM T37693 CGM14Q 25149823 IC50 = 5910 nM T37693 C4H8ZF 25149919 IC50 = 979 nM T37693 C0MAL9 25149920 IC50 = 1120 nM T37693 CX6W8D 25149921 IC50 = 736 nM T37693 CUA60C 25150037 IC50 = 1750 nM T37693 CVS9Y0 25150038 IC50 = 1480 nM T37693 C4RHW0 25150039 IC50 = 407 nM T37693 CO5UQ7 25150040 IC50 = 242 nM T37693 CT02WX 25150041 IC50 > 10000 nM T37693 C8PUM7 25150240 IC50 = 2330 nM T37693 C7E4HJ 25150241 IC50 = 2820 nM T37693 CK94SJ 25150436 IC50 = 1300 nM T37693 CB7QE1 25150437 IC50 = 1810 nM T37693 CW06KG 25150439 IC50 = 375 nM T37693 CSD5M2 25150523 IC50 = 1120 nM T37693 C35BEU 25150524 IC50 = 1670 nM T37693 C9HX6Q 25150527 IC50 = 1890 nM T37693 C16OQZ 25150614 IC50 = 924 nM T37693 C6VL1U 25150616 IC50 = 1050 nM T37693 CU7A2T 25150617 IC50 > 10000 nM T37693 CP0ZF1 25150618 IC50 = 1670 nM T37693 CEPY09 25150619 IC50 = 1730 nM T37693 CO48GN 25150705 IC50 = 539 nM T37693 C8F5KE 25150706 IC50 = 2040 nM T37693 CK15AS 25154780 Ki = 0.9 nM T37693 CYB6T7 25159779 IC50 = 1.95 nM T37693 C9MHD4 25159780 Ki = 91.2 nM T37693 CK3BJ0 25159912 Ki = 120.23 nM T37693 C8IZO3 25159915 Ki = 213.8 nM T37693 CJRM20 25160046 Ki = 257.04 nM T37693 C4V8RQ 25160840 Ki = 5.623 nM T37693 CZ47PT 25168164 Ki > 1000 nM T37693 CMYQ85 25168165 Ki > 1000 nM T37693 C42VOK 25168166 Ki > 1000 nM T37693 C4PKM7 25174143 EC50 = 17 nM T37693 CL9I5F 25178127 Ki = 1000 nM T37693 CK6Z9J 25181419 EC50 = 12.59 nM T37693 CB0F5Z 25181480 EC50 = 5 nM T37693 CWRL74 25181481 EC50 = 25 nM T37693 C9XF6D 25185396 Ki = 21000 nM T37693 C4O3KW 25186235 Ki = 30000 nM T37693 CB8Y1X 25186511 Ki = 1900 nM T37693 CO9Z1E 25194977 IC50 > 10 nM T37693 CDZ2C4 25194999 IC50 > 10 nM T37693 CIE12A 25195000 IC50 > 10 nM T37693 CRW89Y 25195006 EC50 = 17 nM T37693 CX4E8J 25195055 IC50 = 41 nM T37693 CL41UB 25195469 EC50 = 1 nM T37693 C19CNW 25196320 Ki = 26.3 nM T37693 C0MQ7R 25196433 Ki = 49.1 nM T37693 CHS15A 25196434 Ki = 21.5 nM T37693 CR7AX1 25206705 Ki = 20.1 nM T37693 CTL8N0 25211883 EC50 = 11 nM T37693 CO2M3A 25221005 EC50 = 40 nM T37693 CP9Y6Z 25221007 Ki = 177 nM T37693 C4E2ZV 25222459 Ki = 2700 nM T37693 CC9J8H 25222461 Ki = 29.4 nM T37693 CZW14V 25222465 EC50 = 59.1 nM T37693 C2S5OU 25222569 Ki = 127 nM T37693 C5LIC2 25222673 EC50 = 43.6 nM T37693 CJT9H6 25222679 EC50 = 72 nM T37693 CSY93X 25222681 Ki = 144 nM T37693 CKMF58 25223972 Ki = 1020 nM T37693 CAH40Z 25224932 Ki > 10000 nM T37693 C0IXY5 25230443 Ki = 7.1 nM T37693 CF57PX 25230523 Ki = 121 nM T37693 CX8QD0 25256778 Ki = 1.66 nM T37693 CLX7J5 25266053 EC50 = 2 nM T37693 CUNB26 25266054 EC50 = 1 nM T37693 CW5E7B 25266386 EC50 = 62 nM T37693 C5JEQ9 25266387 EC50 = 60 nM T37693 C4Q1WE 25266390 EC50 = 30 nM T37693 CK6E4Y 25266740 EC50 = 180 nM T37693 CKH0D7 25267085 EC50 = 30 nM T37693 CX3RS4 25267089 EC50 = 5 nM T37693 CADY30 25267090 EC50 = 280 nM T37693 C0Q6WY 25267804 EC50 = 60 nM T37693 C6MLV2 25268512 EC50 = 6 nM T37693 CV56WX 25268513 EC50 = 6 nM T37693 CTMD50 25268869 EC50 = 0.51 nM T37693 C3JHI2 25269225 EC50 = 150 nM T37693 CZ02CU 25269919 EC50 = 20 nM T37693 CVLI93 25269921 EC50 > 20000 nM T37693 CGP3A2 25270246 EC50 = 200 nM T37693 CMK28L 25434865 Ki = 120 nM T37693 CCB03W 26123627 EC50 = 4 nM T37693 CI2TB6 26202942 Ki = 10 nM T37693 C1EV6S 26521432 Ki = 540 nM T37693 C0O3XE 26551661 EC50 = 152 nM T37693 C6BKL5 40647161 EC50 = 674 nM T37693 CC50YQ 42596959 Ki = 1000 nM T37693 CU35YL 42601401 IC50 = 386 nM T37693 C1KH3X 42601402 IC50 = 374 nM T37693 C1NKQ6 42605511 IC50 > 5000 nM T37693 CQ2SB1 42605622 IC50 > 1000 nM T37693 CG7M1N 42605623 IC50 > 1000 nM T37693 CY61ZS 42605958 IC50 > 5000 nM T37693 C9TL5Q 42607230 IC50 = 5000 nM T37693 CS4O0I 42607232 IC50 > 5000 nM T37693 CDM67X 42617976 Ki = 23440 nM T37693 CF3HW5 42617977 Ki = 1780 nM T37693 CQ2NR6 42617978 Ki = 6810 nM T37693 CE6T1R 42617980 Ki = 162 nM T37693 C9QF7X 42617987 Ki > 10000 nM T37693 CYB0L5 42617988 Ki > 10000 nM T37693 CW26DC 42617995 Ki = 1258.93 nM T37693 C9P6KA 42617996 Ki = 5011.87 nM T37693 CT2R8P 42625198 Ki = 570 nM T37693 C14VEA 42625199 Ki = 30 nM T37693 CVN5E0 42625200 Ki = 10000 nM T37693 CN4ZG2 42625201 Ki = 199.53 nM T37693 CEYI79 42625202 Ki = 7.9 nM T37693 CV60EY 42625203 Ki = 7.9 nM T37693 C9AK1Y 42625283 Ki = 10000 nM T37693 CZEB13 42625284 Ki = 31.62 nM T37693 CK3J1B 42625285 Ki = 600 nM T37693 CY4WS2 42625463 IC50 > 10000 nM T37693 C64OXN 42625464 IC50 > 10000 nM T37693 CV3FM2 42625548 IC50 > 10000 nM T37693 CZ96KC 42625549 IC50 > 10000 nM T37693 C1U5IS 42625550 IC50 > 10000 nM T37693 C6OKJ2 42625551 IC50 > 10000 nM T37693 C1W2DX 42625635 IC50 > 10000 nM T37693 C9GPZ5 42625636 IC50 > 10000 nM T37693 C4C5QJ 42625708 IC50 > 10000 nM T37693 CJ71PG 42625791 IC50 > 10000 nM T37693 C5XVB9 42625945 IC50 > 10000 nM T37693 C6WYS0 42625946 IC50 > 10000 nM T37693 CHQG38 42625947 IC50 > 10000 nM T37693 CZ4V2A 42625948 IC50 > 10000 nM T37693 C2VA7M 42625949 IC50 > 10000 nM T37693 CQ1YN9 42626020 IC50 > 10000 nM T37693 CIS6H0 42626021 IC50 > 10000 nM T37693 CB18AO 42626022 IC50 > 10000 nM T37693 C7K6PG 42626023 IC50 > 10000 nM T37693 CJ8LY0 42626024 IC50 > 10000 nM T37693 CMDL90 42626165 Ki = 1584.89 nM T37693 CHM37O 42626166 Ki = 158.49 nM T37693 CK27OJ 42626167 Ki = 79.43 nM T37693 CU7MV0 42626168 Ki = 120 nM T37693 C4D9KY 42626169 Ki = 125.89 nM T37693 CT1MQ0 42626170 Ki = 19.95 nM T37693 CL32WK 42626231 Ki = 199.53 nM T37693 C23GWK 42626232 Ki = 31.62 nM T37693 CG9X6Q 42626233 Ki = 510 nM T37693 CH20LC 42626378 Ki = 10000 nM T37693 CW31TV 42626379 Ki = 2420 nM T37693 C6JYX3 43161871 Ki = 200 nM T37693 C2D7FZ 44006806 Ki = 1324.12 nM T37693 CB0FC6 44157583 Ki = 7.9 nM T37693 CLP5D9 44157661 Ki = 70 nM T37693 CZ67SH 44157662 Ki = 1.9 nM T37693 CDT5M6 44157663 Ki = 69.8 nM T37693 CRU08O 44157743 Ki = 3 nM T37693 CFV76H 44157744 Ki = 5.8 nM T37693 C3DW6E 44157745 Ki = 0.7 nM T37693 CVK7D9 44176908 Ki = 26 nM T37693 C8GY4U 44177029 Ki = 2116 nM T37693 CH1XK6 44177030 Ki = 4885 nM T37693 CBCZ24 44177031 Ki = 2928 nM T37693 C56QUX 44177146 Ki = 987 nM T37693 CES0V9 44177147 Ki = 618 nM T37693 CNE39O 44177148 Ki = 918 nM T37693 C34VDU 44177149 Ki = 432 nM T37693 C1NX0K 44177150 Ki = 673 nM T37693 CRE02Z 44177151 Ki = 290 nM T37693 CB2SO4 44177259 Ki = 274 nM T37693 C1V0SA 44177261 Ki = 52 nM T37693 C06NFO 44177371 Ki = 407 nM T37693 CI51QM 44177373 Ki = 329 nM T37693 C9B5WI 44177474 Ki = 356 nM T37693 C32AWN 44177475 Ki = 899 nM T37693 CBZL51 44177476 Ki = 322 nM T37693 CUS85Q 44177477 Ki = 831 nM T37693 C7A3CG 44177478 Ki = 1300 nM T37693 CW3DR7 44177572 Ki = 1043 nM T37693 C70RHS 44177573 Ki = 317 nM T37693 CXS2P1 44191632 IC50 = 1173.7 nM T37693 CA7R6C 44191633 IC50 = 4763.3 nM T37693 CG3K4M 44191634 IC50 = 1950.4 nM T37693 CLU36Q 44191688 IC50 = 2736.6 nM T37693 CCHU94 44191689 IC50 = 768.4 nM T37693 CD50QV 44191690 IC50 = 3968 nM T37693 C36RIL 44191691 IC50 = 1570.6 nM T37693 C10TVJ 44191692 IC50 = 3500.6 nM T37693 CO2FX0 44191743 IC50 = 496.7 nM T37693 CTS48Z 44191747 IC50 = 486.9 nM T37693 CZC56D 44191748 IC50 = 5510.1 nM T37693 CU6RC5 44191749 IC50 = 2881.5 nM T37693 CGY34V 44191806 IC50 = 3177.2 nM T37693 C70DKR 44191807 IC50 = 5126.9 nM T37693 C8PVX1 44191808 IC50 = 7946.1 nM T37693 C4UXE0 44191809 IC50 = 1095.5 nM T37693 C4DGZ9 44191810 IC50 = 1058.5 nM T37693 CIK5H6 44191811 IC50 = 901.4 nM T37693 C5P2OJ 44191879 IC50 = 822 nM T37693 CY0F4D 44191880 IC50 = 10260 nM T37693 CNR43E 44191881 IC50 = 1372.2 nM T37693 CXT7B3 44191882 IC50 = 3249.2 nM T37693 CR7PU3 44191883 IC50 = 4326.9 nM T37693 CMAI32 44191949 IC50 = 4746 nM T37693 CQH87P 44208932 Ki = 0.28 nM T37693 C3QC1N 44222441 Ki > 10000 nM T37693 C56IMC 44227470 EC50 = 1.5 nM T37693 C9L7YS 44227471 EC50 = 0.32 nM T37693 C81ECD 44241663 EC50 = 630.96 nM T37693 COM67A 44241664 EC50 = 794.33 nM T37693 CWA6J4 44247588 Ki > 1000 nM T37693 C8N3DQ 44247599 IC50 = 738 nM T37693 CC32UV 44247671 IC50 > 10000 nM T37693 C45XDC 44247694 IC50 = 488 nM T37693 CDR70U 44248166 Ki = 400 nM T37693 CWC41U 44249869 EC50 = 5.1 nM T37693 C9EYJ3 44249870 EC50 = 7 nM T37693 C6H0GU 44270432 Ki = 1740 nM T37693 CW9LY7 44274794 Ki > 1000 nM T37693 C94SQU 44300691 Ki = 433 nM T37693 CL56ZV 44300702 Ki = 0.58 nM T37693 CRT85E 44300711 Ki = 41.2 nM T37693 CZB85J 44306648 Ki = 2 nM T37693 CS9T4J 44306650 Ki = 110 nM T37693 C76TNB 44307202 Ki = 11 nM T37693 CF8YK9 44307203 Ki = 29 nM T37693 C32MHP 44312382 Ki = 397 nM T37693 C74YBQ 44312424 Ki = 213 nM T37693 C5T8JH 44312516 Ki = 142 nM T37693 C89OGD 44312517 Ki = 27 nM T37693 CP61BT 44312518 Ki = 7840 nM T37693 CP2V5L 44312529 Ki = 8.5 nM T37693 CC68OA 44312599 Ki = 59 nM T37693 C5FWB9 44312617 Ki = 134 nM T37693 CI5NA2 44312651 Ki = 1046 nM T37693 CB72ZP 44312667 Ki = 354 nM T37693 C0AL9Q 44312685 Ki = 14 nM T37693 CUA6G2 44316548 Ki = 120 nM T37693 CHL78P 44316708 Ki = 86 nM T37693 C24SRK 44316743 Ki = 24 nM T37693 CXW9B2 44316762 Ki = 184 nM T37693 CX23MU 44316763 Ki = 8 nM T37693 CT8WA6 44316766 Ki = 22 nM T37693 C1CYS0 44316767 Ki = 71 nM T37693 C86XZQ 44316782 Ki = 263 nM T37693 CHY0V7 44316805 Ki = 205 nM T37693 CKLC83 44316970 Ki = 169 nM T37693 CW8T1H 44316971 Ki = 235 nM T37693 C6PSX3 44317019 Ki = 294 nM T37693 CLYF59 44317079 Ki = 38 nM T37693 C78QDX 44317080 Ki = 20 nM T37693 C9HU1M 44317100 Ki = 41 nM T37693 C5UEJ7 44317113 Ki = 31 nM T37693 C37WXH 44317210 Ki = 30 nM T37693 CP5EN3 44317365 Ki = 251 nM T37693 C6LM9P 44336477 EC50 = 116.2 nM T37693 CSNA89 44339199 Ki = 0.199 nM T37693 CM6T0I 44340976 Ki = 36 nM T37693 CX47WB 44344143 Ki = 0.65 nM T37693 C82CWR 44344222 Ki = 85.9 nM T37693 C8D7CT 44344236 Ki = 17.6 nM T37693 CDKT47 44345983 Ki = 1.023 nM T37693 CKQ25P 44346066 Ki = 0.2884 nM T37693 CPU9G7 44358262 Ki = 1.1 nM T37693 CL3S8T 44388893 Ki = 143 nM T37693 CB3WI0 44388911 Ki = 191 nM T37693 CZVP65 44390375 IC50 > 2000 nM T37693 C9HKY5 44390712 IC50 = 815 nM T37693 CW4CU6 44397424 Ki = 2679 nM T37693 C1IW3H 44397519 Ki = 781 nM T37693 CYJ7C4 44403115 Ki = 1126 nM T37693 C4OT7Z 44403122 Ki = 1871 nM T37693 C5WRH0 44403130 Ki = 2584 nM T37693 C5VZU3 44403136 Ki = 9077 nM T37693 C0A4UK 44404867 Ki = 1.8 nM T37693 C6C1HA 44404868 Ki = 192 nM T37693 CJQ8C2 44404869 Ki = 77 nM T37693 CZ6D4S 44404874 Ki = 16 nM T37693 CPU9T2 44404875 Ki = 230 nM T37693 CGIB02 44404876 Ki = 76 nM T37693 CO3P8E 44404879 Ki = 3.5 nM T37693 CK1D2W 44404880 Ki = 406 nM T37693 CQE37U 44404881 Ki = 35 nM T37693 C6O2CS 44404882 Ki = 86 nM T37693 CLF3M9 44404884 Ki = 2 nM T37693 CBW95T 44404885 Ki = 6 nM T37693 C49UWD 44404890 Ki = 23 nM T37693 CG72OJ 44404891 Ki = 10 nM T37693 CWAR29 44404894 Ki = 128 nM T37693 C45QOF 44404898 Ki = 0.6 nM T37693 CZJ81P 44404903 Ki = 0.9 nM T37693 CU1I5P 44404911 Ki = 232 nM T37693 CJV75P 44404915 Ki = 58 nM T37693 C9JW4R 44404919 Ki = 30 nM T37693 CUX9H5 44404922 Ki = 6 nM T37693 C1O6HS 44404923 Ki = 1.3 nM T37693 CK47QU 44404924 Ki = 410 nM T37693 C4RN7M 44404927 Ki = 0.6 nM T37693 COCU13 44404928 Ki = 6.7 nM T37693 C6J8IT 44404929 Ki = 247 nM T37693 CHE2D0 44404930 Ki = 278 nM T37693 C5YX3O 44404933 Ki = 0.4 nM T37693 C7OBL6 44404934 Ki = 1 nM T37693 CBO36P 44404935 Ki = 983 nM T37693 C1IVU2 44404936 Ki = 164 nM T37693 CVL3S8 44405953 Ki = 4100 nM T37693 CPW2Z0 44405961 Ki = 4000 nM T37693 C91IGO 44405962 Ki = 4200 nM T37693 CMTI01 44405963 Ki > 10000 nM T37693 C49YTQ 44405990 Ki = 5100 nM T37693 C2PMS0 44406005 Ki > 10000 nM T37693 C1OFV8 44406006 Ki > 10000 nM T37693 CPJ3Y5 44406010 Ki > 10000 nM T37693 C1R7KG 44406065 Ki > 10000 nM T37693 C0R8HJ 44406069 Ki > 10000 nM T37693 CDH69R 44406086 Ki > 10000 nM T37693 CIJ4D9 44406096 Ki > 10000 nM T37693 CVK9O1 44406098 Ki > 10000 nM T37693 CJ8DT5 44406099 Ki = 4000 nM T37693 C61TBI 44406108 Ki = 4300 nM T37693 C8UJV2 44406124 Ki > 10000 nM T37693 CRYI42 44406130 Ki > 10000 nM T37693 CH76JQ 44406131 Ki > 10000 nM T37693 CP5OK0 44406141 Ki > 10000 nM T37693 CM4XA8 44406146 Ki = 4000 nM T37693 C0Q2HD 44406147 Ki = 4500 nM T37693 C7RV1K 44406609 EC50 = 14.1 nM T37693 CJ14BS 44406610 Ki = 664 nM T37693 C2O9BM 44406613 Ki = 70.8 nM T37693 C4UHA1 44406629 Ki > 1000 nM T37693 CE8KQ6 44406661 Ki = 174 nM T37693 CEKQ30 44407258 IC50 = 1400 nM T37693 CZW8H2 44407272 IC50 = 1400 nM T37693 C8MA5H 44407369 Ki > 10000 nM T37693 CF7ZB6 44407448 Ki > 10000 nM T37693 CWD09L 44407449 Ki > 10000 nM T37693 CA5G6X 44407528 Ki > 10000 nM T37693 CUF1I7 44407557 Ki > 10000 nM T37693 CP1A5X 44407637 Ki > 10000 nM T37693 C4QK2S 44407664 Ki > 10000 nM T37693 CA59QM 44407775 Ki > 10000 nM T37693 CT34OK 44407776 Ki > 10000 nM T37693 CO2S4P 44407798 Ki > 10000 nM T37693 CY0N7C 44409165 Ki = 51.29 nM T37693 CSD7I2 44409348 Ki = 71.81 nM T37693 CZ7BA2 44409357 Ki = 25.12 nM T37693 CA1P5Z 44409404 Ki = 107.15 nM T37693 C5A3IS 44413438 Ki = 220 nM T37693 CAT37V 44423280 EC50 = 630 nM T37693 CXKZ94 44424074 Ki = 390 nM T37693 CG1W7H 44424075 Ki = 39 nM T37693 C3BV5M 44424076 Ki = 80 nM T37693 CYR36J 44424077 IC50 > 10000 nM T37693 CO14IM 44424078 Ki = 1650 nM T37693 CTIA24 44424079 Ki = 39 nM T37693 CI1NQ7 44424080 Ki = 310 nM T37693 C7G4KI 44424081 Ki = 3940 nM T37693 CES0M4 44424082 Ki = 1800 nM T37693 CGFH81 44424083 Ki = 470 nM T37693 CO29QR 44424084 Ki = 7900 nM T37693 CJ5A9X 44424085 Ki = 2100 nM T37693 CF3WD9 44424086 Ki = 1420 nM T37693 CSGH07 44424087 Ki = 39 nM T37693 C05HAK 44424088 Ki = 280 nM T37693 C3GSH8 44424089 Ki = 2900 nM T37693 CTDP28 44424090 IC50 > 10000 nM T37693 CFV9N7 44424091 IC50 > 10000 nM T37693 C3C5MS 44424092 IC50 > 10000 nM T37693 CFQ5V1 44424093 Ki = 3940 nM T37693 CI27OV 44424094 Ki = 13 nM T37693 C1BI8C 44425206 Ki > 1000 nM T37693 CV2CW6 44425947 IC50 = 284.7 nM T37693 CUZ52I 44425948 IC50 > 2000 nM T37693 C7K3VZ 44425951 IC50 > 2000 nM T37693 CC9S6T 44425955 IC50 = 1441 nM T37693 CE5DV6 44425957 IC50 > 2000 nM T37693 CH31IY 44425960 IC50 = 1488 nM T37693 C50VBY 44425967 IC50 = 668.2 nM T37693 C1RI4V 44425970 IC50 = 807.7 nM T37693 C85WXL 44425974 IC50 = 454.2 nM T37693 C2S4TA 44425977 IC50 = 201.7 nM T37693 C8TW0V 44425983 IC50 = 300.8 nM T37693 C29RVL 44425996 IC50 = 498.2 nM T37693 C3D6XU 44425998 IC50 = 283.5 nM T37693 C8N7SY 44425999 IC50 = 997.8 nM T37693 COY28R 44426001 IC50 > 2000 nM T37693 C7KDN1 44426002 IC50 = 622 nM T37693 CN91SE 44426003 IC50 = 1755 nM T37693 CTE8S2 44426005 IC50 = 1079 nM T37693 C1N8SB 44426006 IC50 = 406 nM T37693 C7BQ6P 44426008 IC50 = 1117 nM T37693 CK1Q6C 44426009 IC50 = 1092 nM T37693 C95NOX 44426010 IC50 > 2000 nM T37693 C8N7RU 44426011 IC50 = 1918 nM T37693 CA4TQ0 44426012 IC50 = 2000 nM T37693 C3YPC6 44426013 IC50 = 1757 nM T37693 CQ7DY8 44426014 IC50 = 904 nM T37693 C5UE3X 44426015 IC50 = 1077 nM T37693 C4BS5C 44426016 IC50 = 1907 nM T37693 C5TJ3O 44426017 IC50 = 180.7 nM T37693 CAO8I2 44426020 IC50 = 945 nM T37693 C4UF8W 44426021 IC50 > 2000 nM T37693 CM7S4D 44426022 IC50 = 1368 nM T37693 CG9ZO2 44426300 Ki = 8300 nM T37693 C04SIN 44426321 Ki = 1100 nM T37693 CQ5L7T 44426373 Ki = 1100 nM T37693 CMTL10 44426375 Ki > 10000 nM T37693 CR9NI6 44426377 Ki = 4000 nM T37693 C5PV6B 44426379 Ki = 3200 nM T37693 C08URI 44426380 Ki = 4500 nM T37693 CJ04FU 44426381 Ki = 6400 nM T37693 CPU6S7 44426382 Ki > 10000 nM T37693 CHEC87 44426383 Ki > 10000 nM T37693 C67YNR 44426384 Ki = 10000 nM T37693 C32KAL 44427439 IC50 = 11000 nM T37693 C9Z3RU 44427440 IC50 = 90 nM T37693 C4AY0T 44427441 IC50 = 85 nM T37693 CUXF91 44427442 IC50 = 660 nM T37693 CWA8H9 44427443 IC50 = 2000 nM T37693 CG4LS0 44427444 IC50 = 120 nM T37693 CPI40O 44431923 Ki = 55 nM T37693 C7GN9T 44431924 Ki = 1.7 nM T37693 CVB6N4 44431929 Ki = 16 nM T37693 C4ADH8 44431933 Ki = 5.6 nM T37693 CY0M2C 44431937 Ki = 14 nM T37693 CS7B0G 44431938 Ki > 1000 nM T37693 CX25NO 44431942 Ki > 1000 nM T37693 C82TOK 44431943 Ki = 600 nM T37693 CVH58M 44431945 Ki = 56 nM T37693 C96LUC 44431947 Ki = 3.6 nM T37693 C9ED7S 44431948 Ki > 1000 nM T37693 CK85UD 44431950 Ki = 140 nM T37693 C6OR5Y 44431952 Ki = 39 nM T37693 C8PR4Q 44431955 Ki = 18 nM T37693 C5PS7M 44431956 Ki = 6.6 nM T37693 CY25PR 44431957 Ki = 20 nM T37693 C3Z4DM 44431958 Ki = 830 nM T37693 C7NWB8 44431960 Ki = 7.8 nM T37693 CRV32B 44431963 Ki = 1700 nM T37693 CP2H7G 44431970 Ki = 45 nM T37693 C0Q6OE 44431973 Ki > 1000 nM T37693 C0BZM8 44431974 Ki > 1000 nM T37693 CGY89J 44431978 Ki = 34 nM T37693 C61GOU 44431987 Ki = 2.3 nM T37693 CX96RE 44431989 Ki = 320 nM T37693 CP7H0J 44431992 Ki > 1000 nM T37693 C87AWH 44431996 Ki = 480 nM T37693 CUY71Q 44432000 Ki = 380 nM T37693 C6PO4R 44432001 Ki > 1000 nM T37693 CW3GF1 44432004 Ki = 660 nM T37693 CJH15F 44432311 Ki = 9 nM T37693 C8Z4HT 44432312 Ki = 65 nM T37693 C8L1GT 44432313 Ki = 1 nM T37693 C5W3KH 44432314 Ki = 2.5 nM T37693 CMC1L8 44432316 Ki = 23 nM T37693 CX84NA 44432317 Ki = 1.1 nM T37693 CPN2C1 44432318 Ki = 1 nM T37693 CUBO91 44432319 Ki = 3.8 nM T37693 CB64PA 44432320 Ki = 1.2 nM T37693 C9RLQ8 44432321 Ki = 7 nM T37693 CZ35SY 44432322 Ki = 18 nM T37693 CW0A7J 44432323 Ki = 2.3 nM T37693 C26SPZ 44432324 Ki = 6.3 nM T37693 CP09WF 44432325 Ki = 1.1 nM T37693 C4EL9R 44432340 Ki = 12 nM T37693 CLR7C4 44432342 Ki = 1 nM T37693 C2FOQ4 44432345 Ki = 5 nM T37693 CW8OK2 44432347 Ki = 0.2 nM T37693 C3EP2D 44432349 Ki = 24 nM T37693 CO7M3T 44432351 Ki = 11 nM T37693 C10FBU 44432352 Ki = 1.3 nM T37693 C5CB6D 44432354 Ki = 0.9 nM T37693 CLQ5E1 44432356 Ki = 1.1 nM T37693 CPOM02 44432708 Ki = 487 nM T37693 C2L9FW 44434974 Ki = 20.3 nM T37693 CO37VG 44434976 Ki = 1.33 nM T37693 CO64PQ 44434993 Ki = 113 nM T37693 C9K6EG 44435004 Ki = 11.7 nM T37693 CP4B1S 44435054 Ki = 371.54 nM T37693 CE2U9J 44435055 Ki = 221.6 nM T37693 C0KUC3 44435059 Ki = 104.71 nM T37693 CGY1K2 44435062 Ki = 109.65 nM T37693 CT2Z7E 44435067 Ki = 50.12 nM T37693 COZ3W7 44435074 Ki = 229.09 nM T37693 C6P7SG 44435076 Ki = 99.23 nM T37693 C9DBI0 44435083 Ki = 32.87 nM T37693 CPTZ16 44435085 Ki = 63.1 nM T37693 CJ47VT 44435574 IC50 = 75 nM T37693 CR57OQ 44435576 IC50 = 170 nM T37693 CE7L1V 44435577 IC50 = 65 nM T37693 CTP6J3 44435579 IC50 = 210 nM T37693 C5HFA8 44435583 IC50 = 490 nM T37693 CI1FE9 44436022 Ki = 83.4 nM T37693 C2F5XE 44436027 Ki = 333 nM T37693 CT67JK 44436028 Ki = 160 nM T37693 CQ4VJ6 44436030 Ki = 221 nM T37693 CNAS45 44436032 Ki = 200 nM T37693 CHLR35 44436034 Ki = 119 nM T37693 CZU01A 44436038 Ki > 4000 nM T37693 C6JIO8 44436039 Ki = 18.2 nM T37693 CC4W9Z 44436043 Ki = 54.6 nM T37693 CQ8OM0 44436044 Ki = 5.3 nM T37693 CUN51T 44436058 Ki = 259 nM T37693 C1EJI5 44436060 Ki = 30.9 nM T37693 C32RIO 44436061 Ki = 23.5 nM T37693 C04YJN 44436063 Ki = 93 nM T37693 CW0YG3 44436066 Ki = 154 nM T37693 C0YK5M 44436067 Ki = 1288 nM T37693 C23ZYX 44436070 Ki > 2000 nM T37693 CIU7D9 44436072 Ki = 1500 nM T37693 CT28WO 44437774 Ki = 78.22 nM T37693 C4T6JW 44437777 Ki = 257.33 nM T37693 CKS32L 44437778 Ki = 10.9 nM T37693 C5UZQ7 44437779 Ki = 7.46 nM T37693 C6RI2M 44437780 Ki = 2.52 nM T37693 CB34DJ 44437781 Ki = 3.13 nM T37693 CE8V6J 44437782 Ki = 189 nM T37693 CM30GA 44440991 IC50 = 320 nM T37693 CW1AG3 44440992 IC50 = 5700 nM T37693 C1W7FC 44440993 IC50 = 2800 nM T37693 CB9AL1 44440994 IC50 = 1800 nM T37693 C75IOU 44440995 IC50 = 4000 nM T37693 CCWQ18 44440996 IC50 = 315 nM T37693 CE3PF2 44440997 IC50 = 2600 nM T37693 CMG6T0 44440998 IC50 = 1100 nM T37693 CH6U8V 44440999 IC50 = 1400 nM T37693 CJ4MX0 44441001 IC50 = 715 nM T37693 CSG2D8 44441002 IC50 = 2100 nM T37693 C3RC0D 44441003 IC50 = 1800 nM T37693 C1A7ZY 44441004 IC50 = 1100 nM T37693 CJTA08 44441005 IC50 = 3700 nM T37693 C4B7IT 44441006 IC50 = 4300 nM T37693 CQN50B 44441007 IC50 = 3300 nM T37693 C8I1UG 44441008 IC50 = 4900 nM T37693 CMO79B 44441009 IC50 = 1600 nM T37693 CABT03 44441010 IC50 = 1800 nM T37693 C7VL0N 44441011 IC50 = 650 nM T37693 C0P4MQ 44441176 Ki = 230 nM T37693 CS9U4H 44441177 Ki = 35 nM T37693 CEH9K8 44441178 Ki = 119 nM T37693 CEWQ75 44441180 Ki = 275 nM T37693 CC5AG8 44441181 Ki > 5000 nM T37693 C6V9ME 44441183 Ki > 5000 nM T37693 C17WNO 44441187 Ki = 915 nM T37693 C4NM8V 44441188 Ki = 1360 nM T37693 C2GKI6 44441189 Ki = 33 nM T37693 CQ7L3C 44441191 Ki = 22 nM T37693 C2PHE0 44441194 Ki = 316 nM T37693 CG17DL 44441195 Ki = 202 nM T37693 CO69UP 44441197 Ki = 54 nM T37693 C8AXY2 44441198 Ki = 57 nM T37693 C23RCZ 44441199 Ki = 313 nM T37693 C0PX8I 44441200 Ki = 252 nM T37693 CRE5X7 44441201 Ki = 722 nM T37693 C1VE2Z 44441202 Ki = 371 nM T37693 C0JWO5 44441203 Ki = 18 nM T37693 C4DB1A 44441204 Ki = 84 nM T37693 CP63AR 44441205 Ki = 141 nM T37693 CRZ4V5 44441206 Ki = 989 nM T37693 CV0NY2 44441207 Ki = 2920 nM T37693 C5DT0G 44441208 Ki > 5000 nM T37693 C43ESH 44441209 Ki = 1581 nM T37693 CC8J5R 44441210 Ki > 5000 nM T37693 CU9LR7 44441211 Ki = 98 nM T37693 CCAK75 44441212 Ki > 5000 nM T37693 CWS7B6 44443136 EC50 = 86 nM T37693 C7A2YG 44443138 IC50 = 20 nM T37693 C2RU3Y 44443139 EC50 = 0.3 nM T37693 CY34UP 44443140 IC50 = 17 nM T37693 C4B3WY 44443141 IC50 = 22 nM T37693 C7Z4NY 44443142 IC50 = 24 nM T37693 CNBC42 44443143 IC50 = 5.7 nM T37693 C7U1DE 44443144 IC50 = 0.5 nM T37693 C3WVB1 44443147 IC50 = 220 nM T37693 C1C0EM 44443148 IC50 = 74 nM T37693 C7HPC4 44443149 IC50 = 46 nM T37693 C6P3MF 44443150 EC50 = 5.6 nM T37693 CZU3M6 44443151 EC50 = 2 nM T37693 C2CZK6 44443152 IC50 = 25 nM T37693 CJKW80 44443153 IC50 = 29 nM T37693 CHB61T 44443154 IC50 = 110 nM T37693 CHX09O 44443155 IC50 = 1000 nM T37693 C0BMK4 44443156 IC50 = 0.41 nM T37693 CD8H4P 44443157 IC50 = 230 nM T37693 C9LE0K 44443158 EC50 = 4 nM T37693 CY14CG 44443159 EC50 = 1.5 nM T37693 CCK4Z5 44443160 EC50 = 2.7 nM T37693 CHVC86 44443161 EC50 = 0.62 nM T37693 CVY34E 44443162 EC50 = 7.3 nM T37693 CH5J7Y 44443368 EC50 = 13.5 nM T37693 C8P2BQ 44443370 EC50 = 15.6 nM T37693 CY69LT 44443371 Ki = 4724 nM T37693 C7RJ8Z 44443372 Ki = 84.7 nM T37693 CJ2KY6 44443373 EC50 = 5 nM T37693 CKB28C 44443375 Ki = 106 nM T37693 C3X6WY 44443379 EC50 = 0.6 nM T37693 C0Y5IS 44443394 EC50 = 1.5 nM T37693 CE5YJ9 44443395 EC50 = 6.7 nM T37693 C4T6WD 44443396 Ki = 88.1 nM T37693 CB4X3O 44443398 EC50 = 1.7 nM T37693 C8U6EH 44443400 Ki = 44.2 nM T37693 CF4J1Q 44443401 Ki = 308 nM T37693 CUHZ49 44443404 Ki = 27.6 nM T37693 CSF47I 44443409 Ki = 107 nM T37693 C68LRJ 44443410 EC50 = 4 nM T37693 CY2EA4 44443414 Ki = 38.1 nM T37693 C6FX1J 44443415 Ki = 27.8 nM T37693 C70JDW 44443417 Ki = 216 nM T37693 CZEH01 44443422 EC50 = 1.7 nM T37693 C9AB0R 44443423 EC50 = 0.3 nM T37693 CZ3NL8 44443425 EC50 = 0.9 nM T37693 C9V7IM 44443426 EC50 = 0.8 nM T37693 C1CJ9Y 44443427 EC50 = 2.7 nM T37693 CK76YZ 44443428 EC50 = 0.5 nM T37693 CAW0S5 44443429 Ki = 935 nM T37693 C3N7TI 44443430 Ki = 1982 nM T37693 CFMQ75 44443432 Ki = 37 nM T37693 CF41HI 44444731 Ki = 94 nM T37693 CDO2Y1 44444732 Ki = 79 nM T37693 C1N2HC 44444733 Ki = 79 nM T37693 CM13FT 44444734 Ki = 6.4 nM T37693 CO40HV 44444735 Ki = 28 nM T37693 C95JLA 44444737 Ki = 7900 nM T37693 CUWH37 44444738 Ki = 790 nM T37693 C9H4MD 44444739 Ki = 1640 nM T37693 CSE7K2 44444740 Ki > 7900 nM T37693 C28XNW 44444741 Ki = 2280 nM T37693 C7IX3A 44444950 Ki = 23.6 nM T37693 C4SXI0 44446802 EC50 = 1 nM T37693 C1AOW6 44446809 EC50 > 20000 nM T37693 CFP2X9 44446810 EC50 = 2 nM T37693 CGK54W 44446811 EC50 = 6 nM T37693 CKM0X1 44446812 EC50 = 18 nM T37693 CYO0N5 44446814 EC50 = 119 nM T37693 CQ4GX7 44446815 EC50 = 5 nM T37693 CQ98KI 44446817 EC50 = 18 nM T37693 CV56YT 44446819 EC50 > 20000 nM T37693 C14JXV 44446829 EC50 = 2 nM T37693 C28YGA 44446831 EC50 = 588 nM T37693 CWC3P8 44446833 EC50 = 4 nM T37693 CF9OM6 44446836 EC50 > 20000 nM T37693 C1B2KA 44448412 EC50 = 4 nM T37693 CNLO42 44448413 EC50 = 1.2 nM T37693 CB3G5Q 44448414 EC50 = 4 nM T37693 CRY47W 44448494 Ki > 10000 nM T37693 CA49WS 44448505 Ki > 10000 nM T37693 C6AY8U 44448506 Ki > 10000 nM T37693 C7ZJ9O 44448536 Ki > 10000 nM T37693 C72IYN 44448539 Ki > 10000 nM T37693 CZTQ62 44448540 Ki > 10000 nM T37693 C4G9YD 44448542 Ki > 10000 nM T37693 CBA36L 44448576 Ki > 10000 nM T37693 CSB9M8 44448577 Ki > 10000 nM T37693 C0J4VA 44448578 Ki > 10000 nM T37693 CGL3J5 44448579 Ki = 8100 nM T37693 COWF13 44448613 Ki = 6200 nM T37693 C7VGI3 44448615 Ki > 10000 nM T37693 CIR53D 44448618 Ki = 5200 nM T37693 CVB6E5 44448647 Ki > 10000 nM T37693 CS9YA3 44448648 Ki > 10000 nM T37693 C7JYR2 44448650 Ki > 10000 nM T37693 C4FXJ0 44449070 EC50 = 125 nM T37693 CRG1Z7 44449071 Ki = 390 nM T37693 CCI20B 44449072 EC50 = 25 nM T37693 C5T0BS 44449073 EC50 = 44 nM T37693 CLG5M9 44449097 EC50 = 21 nM T37693 CYN7U8 44449099 Ki = 8.1 nM T37693 C84CJE 44449124 Ki = 3.9 nM T37693 CQ4X9R 44449155 EC50 = 6.6 nM T37693 C3X6IU 44449157 EC50 = 4.3 nM T37693 CM4O5I 44449158 Ki = 11 nM T37693 C75QPO 44449159 Ki = 3.5 nM T37693 C4YA1F 44449217 Ki = 450 nM T37693 C4U1IW 44449219 Ki = 410 nM T37693 C2GUZ7 44449254 EC50 = 1.2 nM T37693 C3JIT7 44449255 EC50 = 0.5 nM T37693 CO17JQ 44449256 EC50 = 1.6 nM T37693 C3OJ8M 44449259 EC50 = 100 nM T37693 C3Z7YA 44449286 EC50 = 158 nM T37693 C0ZQ5P 44449287 EC50 = 2.5 nM T37693 C6CKG2 44449288 EC50 = 10 nM T37693 CCT6L7 44449317 EC50 = 4 nM T37693 CC6UA9 44449319 EC50 = 1.3 nM T37693 C1C0BX 44449320 EC50 = 1.3 nM T37693 CYQ15R 44449322 EC50 = 1 nM T37693 C6OQW1 44449351 EC50 = 31 nM T37693 C03VHS 44449352 EC50 = 1.6 nM T37693 CT9PX6 44449353 EC50 = 0.8 nM T37693 C2QB5R 44449380 EC50 = 4 nM T37693 CJDF06 44449381 EC50 = 6.3 nM T37693 CH0D6T 44449382 EC50 = 5 nM T37693 C1X4OZ 44449383 EC50 = 125 nM T37693 CN3A4X 44449409 EC50 = 20 nM T37693 CZ9U7S 44449410 EC50 = 4 nM T37693 CBE91D 44449411 EC50 = 20 nM T37693 CT0AL1 44449446 EC50 > 10000 nM T37693 C64RBS 44449449 EC50 = 2000 nM T37693 COCB02 44449472 EC50 < 1 nM T37693 CEZ1N8 44449662 EC50 = 0.8 nM T37693 C6JNS3 44449664 EC50 = 0.4 nM T37693 CVC6K2 44449702 EC50 = 1.2 nM T37693 C8KW6I 44449703 EC50 = 0.8 nM T37693 CHAZ75 44449704 EC50 = 5 nM T37693 C07VOL 44449705 EC50 = 1.6 nM T37693 CZ5SJ4 44449736 EC50 = 0.6 nM T37693 C41HZK 44449738 EC50 = 0.4 nM T37693 C9BI1G 44449739 EC50 = 0.5 nM T37693 C3G5QB 44450408 Ki = 282 nM T37693 C5V3QC 44450418 Ki > 1818.2 nM T37693 C50DPE 44450419 Ki = 1242.8 nM T37693 C2OX1G 44450447 Ki = 194.2 nM T37693 CHC2E3 44452445 Ki > 10000 nM T37693 CK85MY 44452561 Ki = 178 nM T37693 CG40EZ 44452624 Ki > 10000 nM T37693 CH10PO 44452652 EC50 = 1.1 nM T37693 CBJG30 44452653 EC50 = 0.85 nM T37693 C5Z4AM 44452672 Ki > 10000 nM T37693 C76GPX 44452677 EC50 = 0.79 nM T37693 CFR7Y8 44452828 IC50 = 51 nM T37693 C2O9GL 44452870 IC50 = 46 nM T37693 CY03TU 44452894 IC50 = 9.5 nM T37693 CF9VW3 44452896 IC50 = 24 nM T37693 C7A6VS 44452920 IC50 = 300 nM T37693 C81RTH 44452937 IC50 = 1930 nM T37693 CVUZ46 44452961 IC50 = 840 nM T37693 C9VU6D 44452993 IC50 > 10000 nM T37693 C7T2AD 44453099 IC50 = 88 nM T37693 C75KBE 44453101 EC50 = 8.8 nM T37693 CCKA13 44453126 EC50 = 4.4 nM T37693 CJ6B5N 44466638 Ki = 1.199 nM T37693 C8VJ5L 44475188 EC50 = 3302 nM T37693 CO42MQ 44475189 EC50 = 4667 nM T37693 CB93OS 44475190 EC50 = 349 nM T37693 CKL9D6 44475191 EC50 = 48 nM T37693 CZ4E7R 44475345 EC50 = 123 nM T37693 CX8MZ5 44475348 EC50 = 654 nM T37693 CZMG41 44475514 EC50 = 265 nM T37693 CLF27M 44475515 EC50 = 1705 nM T37693 C8TKO9 44475665 EC50 = 145 nM T37693 C4YJ7O 44475667 EC50 = 153 nM T37693 CX9Y5J 44475668 EC50 = 14 nM T37693 CNXU56 44475669 EC50 = 107 nM T37693 C45KSU 44475670 EC50 = 10 nM T37693 C37BCT 44476482 Ki = 584 nM T37693 CJXC18 44476564 Ki > 1000 nM T37693 CMNK07 44476566 Ki = 606 nM T37693 CF6WL7 44476567 Ki > 1000 nM T37693 CO3GJ9 44517703 Ki > 3940 nM T37693 C1YJ6M 44517704 Ki = 2.4 nM T37693 CGXE89 44517762 IC50 = 2960 nM T37693 CGK87Q 44555025 Ki = 305 nM T37693 CV0RU3 44560201 IC50 > 10000 nM T37693 CJKY16 44560203 IC50 > 10000 nM T37693 CL8M3P 44560218 IC50 > 10000 nM T37693 CI0T8G 44560219 IC50 > 10000 nM T37693 C2FCI9 44560231 IC50 > 10000 nM T37693 CFP0N9 44560232 IC50 > 10000 nM T37693 C4D9CJ 44560233 IC50 > 10000 nM T37693 CF2XA9 44560240 IC50 > 10000 nM T37693 CB8T0A 44560241 IC50 = 4820 nM T37693 C7O8DG 44560242 IC50 > 10000 nM T37693 CD05GO 44560243 IC50 > 10000 nM T37693 CL3DV8 44560269 IC50 > 10000 nM T37693 C9W8VR 44560270 IC50 > 10000 nM T37693 C0M2DU 44560271 IC50 > 10000 nM T37693 CT98QB 44560272 IC50 > 10000 nM T37693 C8UBN6 44561004 EC50 = 3.3 nM T37693 CU4SG5 44561005 EC50 = 1 nM T37693 CB25AC 44561006 EC50 = 4.8 nM T37693 CMDC01 44561007 EC50 = 8.3 nM T37693 C71HSJ 44561015 Ki = 13.6 nM T37693 CPTB84 44561045 Ki = 2920 nM T37693 COD91U 44561114 EC50 = 25 nM T37693 CMD3W0 44561115 EC50 = 13 nM T37693 CY36FG 44561116 EC50 = 3.4 nM T37693 C1W9IC 44561150 Ki = 799 nM T37693 C08RTQ 44561151 EC50 = 7.3 nM T37693 CYFN50 44561189 EC50 = 2.4 nM T37693 CK3IH5 44561190 Ki = 526 nM T37693 C9P8KC 44561230 EC50 = 11 nM T37693 CVD07Y 44561231 Ki = 57 nM T37693 CKZS21 44561232 EC50 = 43 nM T37693 C4N9BV 44561233 EC50 = 3.2 nM T37693 C0O2ER 44561273 Ki > 5000 nM T37693 C13COW 44561274 EC50 = 3.2 nM T37693 CPG0S6 44561275 EC50 = 2 nM T37693 CB5S1Y 44561307 EC50 = 3 nM T37693 CG42HW 44561308 EC50 = 22 nM T37693 CD5O4Z 44561342 Ki = 1349 nM T37693 C0EC3G 44561343 EC50 = 2.7 nM T37693 CQDJ15 44561375 EC50 = 2.6 nM T37693 CI18KY 44561376 EC50 = 36 nM T37693 C3N6MT 44561377 EC50 = 2 nM T37693 CFL6K1 44561532 EC50 = 1.3 nM T37693 C1NKS2 44561533 EC50 = 0.52 nM T37693 C80YSF 44561534 EC50 = 1.3 nM T37693 CM1S2X 44561571 EC50 = 1.1 nM T37693 CUH92O 44561572 Ki = 588 nM T37693 C9WP1L 44567376 IC50 > 10000 nM T37693 C85QKG 44567397 IC50 > 10000 nM T37693 CJIT49 44567398 IC50 > 10000 nM T37693 C3WDR4 44567399 IC50 = 4950 nM T37693 CIPL70 44569452 EC50 = 4 nM T37693 C42IGT 44569453 EC50 = 8 nM T37693 C3S9KJ 44569454 EC50 = 19 nM T37693 C1AL6B 44569455 EC50 = 104 nM T37693 CDWS53 44569456 EC50 = 148 nM T37693 C6Y0LF 44569505 EC50 = 33 nM T37693 C9VLE7 44569506 EC50 = 13 nM T37693 C3TO8N 44569507 EC50 = 35 nM T37693 C7CRO4 44569508 EC50 = 57 nM T37693 C91HRZ 44569553 EC50 = 86 nM T37693 CTJR64 44569554 EC50 = 1620 nM T37693 C62ROA 44569555 EC50 > 10000 nM T37693 CX72NB 44569556 EC50 > 10000 nM T37693 CWT7A1 44569557 EC50 = 1300 nM T37693 C9MTC0 44569587 EC50 = 4 nM T37693 CRTA75 44569588 EC50 = 5 nM T37693 CUYD25 44569589 EC50 = 3860 nM T37693 CD6W1Y 44569590 EC50 > 10000 nM T37693 C92FOT 44569622 EC50 = 216 nM T37693 CWQ1K2 44569623 EC50 = 189 nM T37693 CUJ4A1 44569924 EC50 = 398.11 nM T37693 C08SCG 44569925 EC50 = 501.19 nM T37693 CJT9Q2 44569926 EC50 = 398.11 nM T37693 CB5S9R 44569927 EC50 = 50.12 nM T37693 C1HWD3 44570015 EC50 = 79.43 nM T37693 CQ7XA5 44570119 EC50 = 63.1 nM T37693 C5WLK8 44570120 EC50 = 39.81 nM T37693 C1CO2M 44570121 EC50 = 50.12 nM T37693 C34ZJI 44570122 EC50 = 501.19 nM T37693 C1WN9J 44570165 EC50 = 39.81 nM T37693 CM1I9W 44570166 EC50 = 251.19 nM T37693 CCR56A 44570167 EC50 = 398.11 nM T37693 CSE9N3 44570253 EC50 = 1995.26 nM T37693 CX9T2R 44570254 EC50 = 1584.89 nM T37693 CYOA27 44570255 EC50 = 2511.89 nM T37693 CP32DL 44570256 EC50 = 398.11 nM T37693 CB4VL6 44570296 EC50 = 1258.93 nM T37693 C1B0EV 44570522 IC50 > 10000 nM T37693 C27RYN 44570535 EC50 = 63.1 nM T37693 C24JMB 44570559 IC50 > 10000 nM T37693 CQ0P5Y 44570560 IC50 > 10000 nM T37693 CJ8MD3 44570561 IC50 > 10000 nM T37693 C40ZIV 44570573 EC50 = 251.19 nM T37693 CDI76Z 44570574 EC50 = 1000 nM T37693 C3MY6V 44570575 EC50 = 251.19 nM T37693 CT93YR 44570576 EC50 = 398.11 nM T37693 CHR90O 44570577 EC50 = 199.53 nM T37693 C57PTO 44570601 IC50 > 10000 nM T37693 C2Z1WE 44570602 IC50 > 10000 nM T37693 CPHM95 44570603 IC50 > 10000 nM T37693 CVZ47U 44570611 EC50 = 100 nM T37693 CS2G7D 44570612 EC50 = 31.62 nM T37693 C5MIN6 44570613 EC50 = 1584.89 nM T37693 CX7EL4 44570703 IC50 > 1000 nM T37693 CT80RC 44570704 IC50 = 420 nM T37693 CH0UT1 44570766 IC50 = 11 nM T37693 CPT2C6 44570767 IC50 = 123 nM T37693 C5CK0F 44570768 IC50 = 498 nM T37693 CXJN76 44571487 IC50 = 5.9 nM T37693 C5FR4V 44571527 IC50 > 10 nM T37693 C8NDA0 44571528 IC50 > 10 nM T37693 CGA62W 44571564 IC50 > 10 nM T37693 CNBW05 44571566 IC50 > 10 nM T37693 CBV09K 44571567 IC50 > 10 nM T37693 CYLG38 44571593 Ki = 1.5 nM T37693 C68APE 44571594 Ki = 5.8 nM T37693 C13FQU 44571595 Ki = 155 nM T37693 CJQC45 44571596 Ki = 11 nM T37693 CKB8D4 44571640 IC50 > 10 nM T37693 CX16CU 44571641 IC50 > 10 nM T37693 C7TC0V 44571642 IC50 > 10 nM T37693 CBS48G 44571676 Ki = 0.9 nM T37693 C7XF1J 44571677 Ki = 6.8 nM T37693 CKD2R0 44571678 Ki = 1 nM T37693 CCQR65 44571679 Ki = 1 nM T37693 CR10QM 44571680 Ki = 1 nM T37693 C32TAP 44571692 IC50 > 10 nM T37693 C8XGL2 44571725 Ki = 4.7 nM T37693 C0C9FB 44571726 Ki = 0.8 nM T37693 C4JAB8 44571727 Ki = 1.8 nM T37693 CN2T8Z 44571728 Ki = 2.4 nM T37693 C6HM3V 44571773 Ki = 6.6 nM T37693 CJ4AM7 44571774 Ki = 1 nM T37693 C8VM7B 44571775 Ki = 5.8 nM T37693 CC7I1B 44571776 Ki = 1.9 nM T37693 CTJU07 44573418 EC50 = 40 nM T37693 CX6VR9 44573464 EC50 = 615 nM T37693 CLB3Z8 44573542 EC50 > 20000 nM T37693 C6H7BS 44573576 EC50 > 20000 nM T37693 C0D4YR 44573577 EC50 > 20000 nM T37693 CQL80H 44574576 EC50 = 7430 nM T37693 C2LG7H 44574577 EC50 = 15660 nM T37693 CCVH32 44574623 EC50 = 7550 nM T37693 CQ76AC 44574665 IC50 = 1100 nM T37693 CM83FT 44574781 IC50 = 12000 nM T37693 C9TZM7 44574993 IC50 = 18000 nM T37693 CW8RY0 44576567 Ki = 74 nM T37693 C3BA8P 44576568 Ki = 51 nM T37693 CJGC60 44576569 Ki = 484 nM T37693 COC9J6 44576570 Ki = 15 nM T37693 CVI5W4 44576588 Ki = 25 nM T37693 CJ8A9D 44576623 Ki = 20 nM T37693 CU5K7V 44576624 IC50 > 2500 nM T37693 CWJ97V 44576638 IC50 > 2500 nM T37693 CQ7L2J 44576639 Ki = 5 nM T37693 CR14SW 44576640 Ki = 5 nM T37693 CFW4H3 44576641 Ki = 15 nM T37693 CK0G5O 44576652 Ki = 242 nM T37693 C14UVC 44576653 Ki = 338 nM T37693 C93RWF 44576654 Ki = 1 nM T37693 C8EQ0F 44576673 Ki = 92 nM T37693 CQLC63 44576674 Ki = 144 nM T37693 CX6N2C 44576675 Ki = 196 nM T37693 CY94LQ 44576715 Ki > 50000 nM T37693 CNBI92 44576968 EC50 = 8 nM T37693 CEG98D 44576969 EC50 = 0.7 nM T37693 CND4P3 44576970 EC50 = 22 nM T37693 C0SLX2 44577003 Ki = 9 nM T37693 CY0S8V 44577004 Ki = 60 nM T37693 CP5U7C 44577005 IC50 > 1000 nM T37693 C1H6LE 44577006 Ki = 232 nM T37693 CFE0J9 44577551 EC50 = 16 nM T37693 C9GW1T 44577552 EC50 = 3 nM T37693 CJIZ28 44577553 EC50 = 313 nM T37693 C6SC5G 44577607 EC50 = 24 nM T37693 C48TNK 44577700 EC50 = 1780 nM T37693 C3K5WB 44577701 EC50 = 80 nM T37693 C7Q9LK 44577702 EC50 = 1550 nM T37693 CG4A6T 44577703 EC50 = 26 nM T37693 C6TP0R 44577704 EC50 = 1440 nM T37693 CIC7Q0 44578053 EC50 = 2 nM T37693 C26PTA 44578055 EC50 = 1550 nM T37693 CBO9H2 44578091 EC50 = 15 nM T37693 C6G5AM 44578092 EC50 = 50 nM T37693 CC04VP 44578093 EC50 = 465 nM T37693 CD1E4Z 44578094 EC50 = 1600 nM T37693 CX3Y1N 44578140 EC50 = 99 nM T37693 C1ART0 44578141 EC50 = 86 nM T37693 C0HJZ8 44578142 EC50 = 140 nM T37693 CV2ZY7 44578143 EC50 = 376 nM T37693 CL3IQ2 44578212 EC50 = 2860 nM T37693 CJ1MK8 44578213 EC50 = 340 nM T37693 CA5R4C 44578214 EC50 = 19 nM T37693 CKA97I 44578215 EC50 = 32 nM T37693 CD79OE 44578574 Ki = 1400 nM T37693 C7LRN5 44578575 Ki = 290 nM T37693 CD43MU 44578576 Ki = 2300 nM T37693 CBPI67 44578618 Ki > 7900 nM T37693 CFXZ16 44578619 Ki > 7900 nM T37693 C5MY0R 44578620 Ki = 790 nM T37693 C8C5XG 44578653 Ki = 650 nM T37693 C5NFK4 44578654 Ki = 790 nM T37693 CYF2L0 44578655 Ki = 1100 nM T37693 CSX6U1 44578656 Ki = 1200 nM T37693 C6DO8E 44578695 Ki = 2400 nM T37693 C8UP7T 44581023 Ki = 7.2 nM T37693 C7CNY2 44581106 Ki = 342 nM T37693 C0UA7D 44581107 Ki = 23 nM T37693 CT0N5V 44582835 Ki = 5000 nM T37693 CVT0K8 44586998 EC50 = 0.015 nM T37693 CJ38WB 44586999 EC50 = 11 nM T37693 CGK5W6 44587054 EC50 = 110 nM T37693 C9AKC5 44587055 EC50 = 49 nM T37693 C65SDP 44587305 Ki = 5.5 nM T37693 CP6T2X 44588588 Ki = 6400 nM T37693 CHI7K5 44588701 Ki > 10000 nM T37693 C21ZJU 44588702 Ki > 10000 nM T37693 CR1IM7 44591240 Ki = 75 nM T37693 C5P9YH 44591241 Ki = 75 nM T37693 C6N1BV 44591252 EC50 = 25 nM T37693 CGH2M3 44591253 Ki = 11 nM T37693 CH3QA7 44591254 Ki = 14 nM T37693 C1IS0P 44591270 Ki = 23 nM T37693 C6CK0Q 44591271 Ki = 5.2 nM T37693 C5TY6G 44591272 Ki = 5.7 nM T37693 C5OAG4 44591273 Ki = 17 nM T37693 CTN05S 44591293 EC50 = 78 nM T37693 CX3J9M 44591294 Ki > 5000 nM T37693 CI4F5K 44591295 EC50 = 64 nM T37693 CU2Z1B 44591296 Ki = 27 nM T37693 CB87ZC 44591297 Ki = 100 nM T37693 CZC2V8 44591328 Ki = 36 nM T37693 C0RG5Z 44591329 Ki = 23 nM T37693 C8EZ2F 44591330 Ki = 81 nM T37693 CFJ6T4 44591331 Ki = 59 nM T37693 C9VER2 44591332 EC50 = 110 nM T37693 CB92EJ 44591350 Ki = 87 nM T37693 C2VMW7 44591351 EC50 = 130 nM T37693 C5MY2H 44591352 Ki = 9.4 nM T37693 CIZR27 44591353 Ki = 11 nM T37693 C1GB8U 44591372 EC50 = 33 nM T37693 COL9S4 44591395 Ki = 660 nM T37693 CE6FA1 44591396 Ki = 2000 nM T37693 CW4DJ1 44592049 Ki > 10000 nM T37693 CIB17U 44592050 Ki >= 10000 nM T37693 C0PLI4 44592051 Ki >= 10000 nM T37693 CYCD37 44592052 Ki > 10000 nM T37693 CC2K9Z 44592083 Ki = 2160 nM T37693 CUP07N 44592084 Ki = 4760 nM T37693 C04SGM 44592085 Ki = 1540 nM T37693 C0NJE8 44592106 Ki = 13.6 nM T37693 C8LM6U 44592114 Ki = 9390 nM T37693 C3TF4I 44592115 Ki = 5240 nM T37693 C5WG4Z 44592116 Ki = 3370 nM T37693 C2FO0R 44592149 Ki = 2780 nM T37693 CUJ3G1 44592150 Ki = 3650 nM T37693 CZKO56 44592151 Ki = 5670 nM T37693 C8NR3G 44592191 Ki > 10000 nM T37693 C0QE1U 44592192 Ki > 10000 nM T37693 CT3W9C 44592193 Ki > 10000 nM T37693 C8JZ2L 44592194 Ki > 10000 nM T37693 CQ45LI 44593416 Ki = 2.53 nM T37693 CU5QM9 44593417 Ki = 0.91 nM T37693 CUS0P8 44593426 Ki = 10.65 nM T37693 C96SDI 44593427 Ki = 7.45 nM T37693 CALE39 44593428 Ki = 0.67 nM T37693 COX3D7 44593429 Ki = 7.83 nM T37693 C3LH5A 44593430 Ki = 12.4 nM T37693 C6URQ2 44593432 Ki = 1.54 nM T37693 C6AKT4 44593433 Ki = 0.54 nM T37693 CC0ZX7 44593612 Ki = 5 nM T37693 CS16LT 44608360 Ki > 1000 nM T37693 CH3K4A 44608519 Ki > 1000 nM T37693 CU26YR 44608681 Ki > 1000 nM T37693 CW9TR0 44608682 Ki > 1000 nM T37693 CMC89D 44626286 Ki = 318 nM T37693 CL25CW 44626287 Ki = 571 nM T37693 CMS21C 44626293 Ki = 247 nM T37693 CW62LE 44626508 Ki > 1000 nM T37693 CHCX20 44626509 Ki > 1000 nM T37693 CWH62A 44626510 Ki > 1000 nM T37693 CF98KL 44626511 Ki > 1000 nM T37693 C4HA1P 44626512 Ki = 1 nM T37693 CP5D3I 44626513 Ki = 9.12 nM T37693 CHQ34G 44626514 Ki = 1.995 nM T37693 CYB13E 44626619 Ki = 1.8 nM T37693 CLI40Y 44626620 Ki > 1000 nM T37693 C57FZK 44626621 Ki = 2.9 nM T37693 CJLY69 44626623 Ki > 1000 nM T37693 C9VP2H 44626624 Ki = 30 nM T37693 CM5Q6F 44626625 Ki = 3.631 nM T37693 C56HJF 44626626 Ki = 68 nM T37693 CQ9ZE1 44626729 Ki = 190 nM T37693 CQ90WV 44626834 Ki = 5.8 nM T37693 CY4UX7 44627979 EC50 = 819 nM T37693 CN01CV 44627980 EC50 = 86 nM T37693 CONU92 44627981 Ki = 15.85 nM T37693 CVCP89 44627983 EC50 = 716 nM T37693 CH1S3P 44627984 Ki = 34.67 nM T37693 CL2PS3 44628086 Ki = 10.96 nM T37693 C4VB5F 44628087 Ki = 2.57 nM T37693 CP2Y8T 44628090 Ki > 1000 nM T37693 CAL60M 44629129 Ki = 219 nM T37693 CN91XU 44806719 Ki > 10000 nM T37693 CD0B8E 45101490 IC50 = 353 nM T37693 C2TYD1 45254043 Ki = 2.7 nM T37693 C7QW2B 45256133 EC50 = 11 nM T37693 CYU95D 45256135 EC50 = 0.66 nM T37693 CUF51H 45266954 Ki = 6.501 nM T37693 C28LNV 45266978 Ki = 9.594 nM T37693 CP04HQ 45267006 Ki = 3.802 nM T37693 C83IUH 45267042 Ki = 10 nM T37693 C0OMI4 45267043 Ki = 10.5 nM T37693 CYDB14 45267487 EC50 = 2511.89 nM T37693 CCES19 45267777 EC50 = 560 nM T37693 CS5LX7 45267778 EC50 = 3000 nM T37693 C3L8NF 45267819 Ki = 14 nM T37693 CUC6B4 45267820 Ki = 0.7295 nM T37693 CMR4S2 45267825 Ki = 440.55 nM T37693 CN41VA 45267831 Ki = 123.03 nM T37693 C8VQ4O 45267840 Ki = 5.598 nM T37693 C80TWH 45268581 EC50 = 295 nM T37693 CGZ27K 45268648 EC50 = 380 nM T37693 C8PN1K 45268654 EC50 = 637 nM T37693 CR1ST7 45268702 Ki = 1.099 nM T37693 C7IH9P 45268706 Ki = 11.99 nM T37693 CR28GB 45268707 Ki = 0.4198 nM T37693 CV52ED 45268709 Ki = 239.88 nM T37693 CK5F2O 45268712 Ki = 25 nM T37693 CIDM75 45269488 EC50 = 21.5 nM T37693 C4YU2C 45269498 EC50 = 320 nM T37693 CJ8EZ5 45269504 EC50 = 9.1 nM T37693 CBVE04 45269512 EC50 = 14.2 nM T37693 CW1KE5 45269566 Ki = 11.99 nM T37693 CW0LY5 45270326 EC50 = 13.4 nM T37693 CC1DS6 45270335 EC50 = 523 nM T37693 C76EPY 45270342 EC50 = 7.9 nM T37693 CB50KY 45270383 Ki = 105.93 nM T37693 CC60PR 45270396 Ki = 0.6902 nM T37693 CB37SM 45270408 Ki = 73.96 nM T37693 C9AXR8 45270409 Ki = 220.8 nM T37693 C16OZV 45271160 EC50 = 1020 nM T37693 C8HCG1 45271208 Ki = 169.82 nM T37693 C2ZES0 45271217 Ki = 6.902 nM T37693 CDQ16L 45271218 Ki = 70.96 nM T37693 CJ03EQ 45271228 Ki = 52 nM T37693 CSY63A 45271747 EC50 = 501.19 nM T37693 C3H6PI 45272056 EC50 = 26.7 nM T37693 CNA9C8 45272115 Ki = 97.05 nM T37693 C50KRU 45272116 Ki = 1.901 nM T37693 C6Y5GS 45272119 Ki = 10.4 nM T37693 C4CXU8 45272121 Ki = 0.6 nM T37693 CPSY23 45272127 Ki = 48.98 nM T37693 CTX4B5 45272618 EC50 = 3162.28 nM T37693 CR14DO 45272684 EC50 = 1995.26 nM T37693 CBXC51 45272685 EC50 = 2511.89 nM T37693 C1YC7M 45272871 EC50 = 21.8 nM T37693 CNX7Y8 45272883 EC50 = 403 nM T37693 CJK2T4 45272898 EC50 = 55.4 nM T37693 CIY0N9 45272899 EC50 = 18.5 nM T37693 CG52KE 45272906 EC50 = 878 nM T37693 CK1G9C 45272969 Ki = 7.194 nM T37693 C2T9IU 45273608 EC50 = 1995.26 nM T37693 CWU0H8 45273822 EC50 = 439 nM T37693 C18TBE 45273832 EC50 = 24.5 nM T37693 CAMX32 45277748 Ki = 526 nM T37693 C6UVZ0 45277749 Ki = 25 nM T37693 CK5G2I 45277750 Ki = 159 nM T37693 C8Y6OP 45375860 IC50 = 38.5 nM T37693 CMO74A 45375898 EC50 = 100 nM T37693 CKW5H7 45375900 EC50 = 79.43 nM T37693 C2P7DZ 45482145 Ki = 20 nM T37693 CI2L3H 45482146 Ki = 100 nM T37693 C2RHP4 45482154 Ki = 80 nM T37693 C5AYP0 45482155 Ki > 3940 nM T37693 CLY7J6 45482156 Ki > 3940 nM T37693 CVX13E 45482170 Ki = 940 nM T37693 CLD6B9 45482181 Ki = 609 nM T37693 CN2D1B 45482194 Ki > 3940 nM T37693 CP3A2G 45482195 Ki = 553 nM T37693 CS8IL1 45482196 Ki > 3940 nM T37693 CRZ7E0 45482212 Ki > 3940 nM T37693 C83GHF 45482213 Ki > 3940 nM T37693 CPB4V3 45482221 Ki = 2887 nM T37693 CKZD49 45482222 Ki = 3483 nM T37693 C5V0BJ 45482230 Ki > 3940 nM T37693 CDI5R8 45482231 Ki = 310 nM T37693 CC1N8T 45482236 Ki > 3940 nM T37693 C71YGP 45482237 Ki = 170 nM T37693 CD8O6R 45482242 Ki = 80 nM T37693 C3FZ2G 45482253 Ki = 790 nM T37693 CJS5B4 45482262 Ki > 3940 nM T37693 C4BMX6 45482263 Ki = 790 nM T37693 C0KX7R 45482264 Ki = 1291 nM T37693 C69UKE 45482265 Ki = 1945 nM T37693 C0SW4I 45482271 Ki > 3940 nM T37693 C3WO9A 45482272 Ki = 667 nM T37693 C01KMJ 45482275 Ki = 12 nM T37693 CMZI72 45482276 Ki = 4.2 nM T37693 CY2C1A 45482277 Ki > 3940 nM T37693 CU2A6Y 45482278 Ki = 3400 nM T37693 C97TZR 45482285 Ki = 1200 nM T37693 C0RK2J 45482286 Ki = 12 nM T37693 CMLT59 45482287 Ki = 373 nM T37693 C8YK5V 45482288 Ki > 3940 nM T37693 CM1QD0 45482290 Ki = 1.3 nM T37693 CB9F2E 45482291 Ki = 20 nM T37693 C9QCD0 45482292 Ki = 1.6 nM T37693 CLM52Q 45482293 Ki = 1100 nM T37693 CG8ME6 45482294 Ki = 12 nM T37693 CE0C1R 45482295 Ki > 3940 nM T37693 C1IUF2 45482296 Ki = 721 nM T37693 C9NPK7 45482298 Ki = 200 nM T37693 CGDH61 45482299 Ki = 900 nM T37693 C8CNJ6 45482300 Ki = 110 nM T37693 C3CJY6 45482302 Ki = 5.7 nM T37693 CX1W2E 45482305 Ki = 739 nM T37693 CV2H0Q 45482306 Ki > 3940 nM T37693 C7WH3G 45482308 Ki > 3940 nM T37693 CF5AU0 45482309 Ki > 3940 nM T37693 CT61ZB 45482312 Ki > 3940 nM T37693 CI4KQ8 45484652 Ki = 8.6 nM T37693 C80ZSJ 45484668 Ki = 19 nM T37693 CWO0Z4 45484669 Ki = 17 nM T37693 C7VJO3 45484677 Ki = 37 nM T37693 CX3HS0 45484683 Ki = 120 nM T37693 C0US3O 45484688 Ki = 45 nM T37693 C93GPE 45484689 Ki = 62 nM T37693 CC8AR5 45484690 Ki = 440 nM T37693 CG5KM4 45484698 Ki = 300 nM T37693 CR8OU6 45484699 Ki = 83 nM T37693 CQ9E8H 45484714 Ki = 700 nM T37693 C1TH8B 45484715 Ki = 1200 nM T37693 CYVW54 45484720 EC50 = 500 nM T37693 C4ENV9 45484721 Ki = 2.3 nM T37693 CS4Z1M 45484728 EC50 = 14 nM T37693 C9IS4Y 45484737 Ki = 70 nM T37693 COE72V 45484738 EC50 = 110 nM T37693 C0L4KU 45484747 Ki = 3.9 nM T37693 CPO14R 45486125 IC50 = 427 nM T37693 CTW7R1 45486126 IC50 > 10000 nM T37693 CMF4A0 45486154 IC50 = 414 nM T37693 CQG4D2 45486165 EC50 = 63.1 nM T37693 C0VYP1 45486166 EC50 = 39.81 nM T37693 C3BN5R 45486180 EC50 = 100 nM T37693 C95TXR 45486181 EC50 = 316.23 nM T37693 C9WL0M 45486183 EC50 = 10000 nM T37693 C2HI9W 45486185 EC50 = 501.19 nM T37693 C43WIN 45486186 EC50 = 398.11 nM T37693 C8PO1D 45486188 EC50 = 501.19 nM T37693 C79HNB 45486189 EC50 = 158.49 nM T37693 C8RFV1 45486191 EC50 = 251.19 nM T37693 CQ83YO 45486193 EC50 = 794.33 nM T37693 CD2I1T 45486194 EC50 = 1258.93 nM T37693 CGMD63 45486195 EC50 = 1000 nM T37693 CA40VN 45486196 EC50 = 251.19 nM T37693 CT64HQ 45486197 EC50 = 79.43 nM T37693 CV06UY 45486198 EC50 = 3981.07 nM T37693 C8RXB2 45486199 EC50 = 2511.89 nM T37693 CNKE85 45486200 EC50 = 1584.89 nM T37693 C8CR2E 45486201 EC50 = 125.89 nM T37693 C6M5BV 45486202 EC50 = 63.1 nM T37693 C68SFQ 45486204 EC50 = 1000 nM T37693 CIE6R2 45486207 EC50 = 794.33 nM T37693 CBF0J3 45486209 EC50 = 398.11 nM T37693 CZ5EP0 45486213 EC50 = 501.19 nM T37693 CQ2JO9 45486214 EC50 = 630.96 nM T37693 C7TQB2 45486215 EC50 = 79.43 nM T37693 C4MR0N 45486216 EC50 = 251.19 nM T37693 C5DOQ2 45486217 EC50 > 31622.78 nM T37693 CRE78C 45486220 EC50 > 31622.78 nM T37693 CT7D5W 45486221 EC50 = 3981.07 nM T37693 C9PR0W 45486227 EC50 = 6309.57 nM T37693 C0R2LC 45486228 Ki = 22.39 nM T37693 C5XH8U 45486229 Ki = 8.3 nM T37693 CF7DI2 45486232 Ki = 2.1 nM T37693 C5MGW3 45486233 Ki = 5.888 nM T37693 C28VPU 45486235 Ki = 154.88 nM T37693 CMS0L5 45486237 Ki > 1000 nM T37693 C93XDH 45486386 Ki > 1000 nM T37693 CX42VA 45486394 Ki = 571 nM T37693 CNDU21 45486467 Ki > 1000 nM T37693 CG9D2X 45486479 Ki > 1000 nM T37693 CBL5Q4 45486480 Ki > 1000 nM T37693 CNE83F 45486585 IC50 = 3863 nM T37693 CL7O8R 45486588 IC50 = 419 nM T37693 CL2M1O 45486624 IC50 = 322 nM T37693 CZI3A7 45486625 IC50 = 699 nM T37693 CDZ06Y 45486626 IC50 = 547 nM T37693 C5LM1E 45486627 IC50 = 1830 nM T37693 CFU06M 45486645 IC50 = 14020 nM T37693 CX03TG 45487312 IC50 = 117 nM T37693 CO02JA 45487319 IC50 = 3213 nM T37693 CR31BT 45487337 IC50 = 5158 nM T37693 C4RWJ7 45487338 IC50 = 25890 nM T37693 C1HX4V 45487344 IC50 = 254 nM T37693 CDME83 45487345 IC50 = 1721 nM T37693 CQ48YZ 45487350 IC50 = 2312 nM T37693 C6MSZ4 45487367 IC50 = 234 nM T37693 C6QZT8 45487368 IC50 = 6113 nM T37693 CYID78 45487377 IC50 = 13290 nM T37693 CV8Y7U 45487389 IC50 = 1414 nM T37693 CC5WX3 45487684 Ki = 13 nM T37693 CA6JH8 45487685 Ki = 7 nM T37693 CJC8B3 45487735 EC50 = 504 nM T37693 CA7H4J 45487736 EC50 = 188 nM T37693 CM07ZR 45487750 Ki = 100 nM T37693 C5BD3E 45487753 EC50 = 15 nM T37693 C8JTA9 45487760 Ki = 870 nM T37693 CACM89 45487771 Ki = 81 nM T37693 CXA9P3 45487780 Ki = 5.3 nM T37693 CK25FM 45487781 Ki = 63 nM T37693 CSW1O4 45487782 Ki = 45 nM T37693 C82GUQ 45504069 Ki = 1060 nM T37693 CN31HO 46191641 EC50 = 50.12 nM T37693 CME02J 46209990 IC50 = 5 nM T37693 C0JCR7 46210310 Ki = 50.5 nM T37693 CS81HE 46216704 Ki > 2220 nM T37693 C4SD8K 46216705 Ki = 1384 nM T37693 C8TFL3 46216706 Ki = 1578 nM T37693 C2VP6F 46216778 Ki = 1407 nM T37693 CW4E2J 46220521 EC50 = 8.8 nM T37693 CYQ03E 46224624 Ki = 14 nM T37693 C3R0TH 46224630 Ki = 9 nM T37693 CDS69K 46224634 Ki = 94 nM T37693 C5PKX3 46224635 Ki = 8.4 nM T37693 CFM82X 46224639 Ki = 90 nM T37693 C1UNT4 46224640 Ki = 66 nM T37693 C4TVW9 46224645 Ki = 760 nM T37693 CCIT36 46224654 Ki = 43 nM T37693 C97HOB 46224658 Ki = 410 nM T37693 CS5TO6 46224659 Ki = 6.9 nM T37693 C7X2AF 46224661 Ki = 12 nM T37693 CBOD08 46224662 Ki = 2.7 nM T37693 C6D5UP 46226066 EC50 > 31622.78 nM T37693 C65MPA 46226067 EC50 = 1584.89 nM T37693 CC2Y3O 46226068 EC50 = 7943.28 nM T37693 CH9V2M 46226069 EC50 = 1258.93 nM T37693 C18GLZ 46226070 EC50 = 12589.25 nM T37693 CL0KM4 46226071 EC50 = 1258.93 nM T37693 C3UFW0 46226083 EC50 = 1000 nM T37693 C1Y2ZD 46226084 EC50 = 1995.26 nM T37693 C54MRO 46226085 EC50 = 158.49 nM T37693 C97WVQ 46226086 EC50 = 398.11 nM T37693 CXA8H5 46226087 EC50 > 31622.78 nM T37693 C3KQY6 46226088 Ki = 2950 nM T37693 CD07HW 46226089 Ki = 234 nM T37693 C9M4EP 46226090 Ki = 43 nM T37693 C58RHI 46226108 EC50 > 31622.78 nM T37693 CR97PI 46226109 EC50 > 31622.78 nM T37693 C63IRS 46226110 EC50 = 630.96 nM T37693 CAP1I4 46226111 EC50 > 31622.78 nM T37693 C64NOG 46226112 EC50 = 251.19 nM T37693 CDH3B0 46226113 EC50 = 158.49 nM T37693 CNV75F 46226114 Ki = 180 nM T37693 C4L2HM 46226115 Ki = 92 nM T37693 CMDO26 46226116 Ki = 750 nM T37693 CDS2G6 46226147 EC50 = 199.53 nM T37693 CVJF51 46226148 EC50 = 79.43 nM T37693 CSI65H 46226149 EC50 = 39.81 nM T37693 CWU43D 46226150 Ki = 1.5 nM T37693 C1D3FQ 46226151 Ki = 7 nM T37693 C6L4PR 46226152 Ki = 8 nM T37693 CHCT54 46226167 Ki = 0.2 nM T37693 CJ7T4D 46226168 Ki = 5.4 nM T37693 CGR9I8 46226169 Ki = 21 nM T37693 C6KER3 46226224 Ki = 3 nM T37693 CAH58K 46226225 Ki = 5.1 nM T37693 C53ODR 46226226 Ki = 37.5 nM T37693 CLG0E3 46226227 Ki = 2460 nM T37693 C0W9DL 46226238 Ki = 202.5 nM T37693 CNG98O 46226239 Ki = 350 nM T37693 CP8U5O 46226240 Ki = 1.1 nM T37693 C8NIK4 46226256 Ki = 1.6 nM T37693 CIL85Q 46226257 Ki = 0.65 nM T37693 CRJ5F7 46226258 Ki = 2 nM T37693 CCQ19F 46226276 Ki = 5 nM T37693 CAK5M4 46226277 Ki = 3 nM T37693 CQ6L5E 46226278 Ki = 0.9 nM T37693 CH79SZ 46226402 EC50 = 199.53 nM T37693 CHA43R 46226403 EC50 = 39.81 nM T37693 CSAC85 46226404 EC50 = 79.43 nM T37693 C14LTF 46226405 EC50 = 39.81 nM T37693 CT6KI2 46226406 EC50 = 50.12 nM T37693 CZS4L3 46226407 EC50 = 100 nM T37693 CC5YA2 46226408 EC50 = 6.31 nM T37693 CS79CQ 46226425 EC50 = 15.85 nM T37693 CGWY69 46226426 EC50 = 630.96 nM T37693 C5JDX0 46226427 EC50 = 25.12 nM T37693 CA9NO8 46226428 EC50 = 1.259 nM T37693 CR7K0F 46226429 EC50 = 0.631 nM T37693 CXA5W9 46226430 EC50 = 199.53 nM T37693 CEXZ31 46227715 Ki = 40 nM T37693 C27OTR 46227717 Ki = 2080 nM T37693 CVI51K 46227718 Ki = 110 nM T37693 CC29JS 46227721 Ki = 6.6 nM T37693 CV7H3L 46227722 Ki = 17 nM T37693 C3OG7F 46227727 Ki = 9.7 nM T37693 CIH45R 46227729 Ki = 1.1 nM T37693 CR8H5M 46227730 Ki = 290 nM T37693 C67KXM 46227739 Ki = 16 nM T37693 C6GY9H 46227741 Ki = 120 nM T37693 CPJ43K 46229257 Ki = 27.95 nM T37693 C34LAI 46229258 Ki = 496.7 nM T37693 CTA7F0 46229282 Ki = 1008 nM T37693 CY7JA8 46229283 Ki = 1068 nM T37693 C6E5BK 46229284 Ki = 1330 nM T37693 C4GEX6 46229285 Ki = 23.8 nM T37693 CIF9G1 46229732 Ki = 574 nM T37693 CNQ71K 46229733 Ki > 1778 nM T37693 C6UFE7 46229734 Ki > 1765 nM T37693 COG0D9 46229778 Ki > 1846 nM T37693 CEO0H4 46229779 Ki > 1678 nM T37693 CW9NS3 46229780 Ki > 1846 nM T37693 C8OCJ7 46229781 Ki > 1846 nM T37693 C0H1NZ 46229782 Ki > 1846 nM T37693 CTD56S 46229826 Ki = 1846 nM T37693 CQ9UG4 46229828 Ki > 1847 nM T37693 CM2L5W 46229864 Ki > 1847 nM T37693 CR7CP6 46229896 Ki > 2220 nM T37693 CF6P0K 46229897 Ki > 2220 nM T37693 C7A9XG 46229898 Ki > 2220 nM T37693 CWF2G6 46229969 Ki > 2400 nM T37693 C5YE2W 46229970 Ki > 2450 nM T37693 CV8O4J 46229971 Ki > 2400 nM T37693 CI36WU 46230014 Ki > 1846 nM T37693 C2TPH4 46230015 Ki > 2000 nM T37693 C4FVX8 46230016 Ki > 1846 nM T37693 C59CRV 46230017 Ki > 2222 nM T37693 CV6KM4 46230070 Ki > 1846 nM T37693 C6W3YJ 46230071 Ki > 2400 nM T37693 CW3Z1X 46230072 Ki > 1500 nM T37693 CSZ9L3 46230073 Ki = 1578 nM T37693 CU7KB8 46230122 Ki = 368 nM T37693 C5ZC0J 46230123 Ki = 1384 nM T37693 CDVT81 46230124 Ki = 368 nM T37693 C6J5SC 46230125 Ki = 1846 nM T37693 CE52LR 46230610 IC50 = 3510 nM T37693 C1GS2E 46230647 IC50 = 3330 nM T37693 C7Y3CB 46230705 IC50 = 6480 nM T37693 C3UI7A 46230816 IC50 = 1790 nM T37693 CUQY29 46230817 IC50 = 2420 nM T37693 CCV73D 46230868 IC50 = 4060 nM T37693 C1JY6B 46230869 IC50 = 3200 nM T37693 CU3MI5 46230870 IC50 = 2570 nM T37693 CDW1O9 46230974 EC50 = 158.49 nM T37693 CK31LV 46230975 Ki = 20 nM T37693 C34LDI 46231031 EC50 = 7.943 nM T37693 CNW5V6 46231032 EC50 = 5.012 nM T37693 CB1OC6 46231088 EC50 = 1.585 nM T37693 C6FAH7 46231089 EC50 = 6.31 nM T37693 CL17TN 46231164 Ki = 50 nM T37693 C18GER 46231255 IC50 = 296 nM T37693 CI3LY6 46231256 IC50 = 582 nM T37693 C4EI1G 46231257 IC50 = 547 nM T37693 CWZ70O 46232373 Ki = 2190 nM T37693 CMZ9G4 46232374 Ki = 1260 nM T37693 C8E0NF 46232375 Ki = 1210 nM T37693 CKX9T8 46232376 Ki > 3000 nM T37693 C7SAY6 46232377 Ki = 2000 nM T37693 CP6D1J 46232431 Ki = 215 nM T37693 C6O8JZ 46232432 Ki = 387 nM T37693 CZ1H6V 46232433 Ki = 1400 nM T37693 C9AOF0 46232434 Ki = 1720 nM T37693 CV02TB 46232435 Ki > 3000 nM T37693 CHE64C 46232505 Ki = 2050 nM T37693 CU36FE 46232506 Ki = 1400 nM T37693 C9UO1G 46232507 Ki > 3000 nM T37693 C30YXI 46232508 Ki = 1770 nM T37693 CZA8J2 46232547 Ki > 3000 nM T37693 CLI29U 46232548 Ki > 3000 nM T37693 CF8D6Z 46232549 Ki > 3000 nM T37693 CT02GZ 46232550 Ki = 782 nM T37693 CC58RP 46232551 Ki = 1500 nM T37693 C3OYB9 46232577 Ki = 469 nM T37693 CNML95 46232578 Ki = 1930 nM T37693 CL0S8C 46232579 Ki = 0.2 nM T37693 C5Y8LD 46232580 Ki = 5.3 nM T37693 CCU94R 46232610 Ki = 2.9 nM T37693 CTYP68 46232611 Ki = 216 nM T37693 C6QGB3 46232612 Ki = 257 nM T37693 COKU52 46232613 Ki = 1090 nM T37693 CS6UC7 46232638 Ki = 255 nM T37693 CA94OK 46233073 Ki > 3000 nM T37693 C6B5LZ 46239964 EC50 = 0.04 nM T37693 C5G3VL 46309339 Ki = 1580 nM T37693 C9IKL7 46833780 EC50 = 20 nM T37693 CSX30A 46834060 EC50 = 22.8 nM T37693 CCT97N 46843358 EC50 = 34 nM T37693 CNM5O6 46843431 EC50 = 6.1 nM T37693 CC07EJ 46843432 EC50 = 6.1 nM T37693 CV03HY 46843437 EC50 = 1150 nM T37693 C52SRT 46843872 EC50 = 5000 nM T37693 CN6M3Y 46851728 EC50 = 14 nM T37693 C7DYR8 46851729 EC50 = 13 nM T37693 C56HDV 46851886 EC50 = 5.9 nM T37693 C43ZMW 46852048 EC50 = 40 nM T37693 CK8N2W 46852211 EC50 = 16 nM T37693 CD04SA 46852212 EC50 = 19 nM T37693 C8QFK3 46852213 EC50 = 7.7 nM T37693 CA9PE1 46852366 EC50 = 14 nM T37693 C2QA8S 46856243 EC50 = 25 nM T37693 C0J1EU 46856244 EC50 = 5 nM T37693 CY3CE6 46861579 EC50 = 0.09 nM T37693 CE2R3U 46869263 Ki = 317 nM T37693 C94EJG 46869398 EC50 = 38 nM T37693 C97JEP 46871671 IC50 = 2260 nM T37693 CFV3T7 46871949 EC50 = 10.5 nM T37693 CPAK05 46872381 EC50 = 329 nM T37693 C95GAX 46872383 EC50 = 19 nM T37693 C8INY3 46872497 EC50 = 15 nM T37693 CK75SZ 46872613 EC50 > 1000 nM T37693 CQNL15 46873104 EC50 = 416 nM T37693 CEZ42W 46873105 EC50 > 1000 nM T37693 C2F1LZ 46873202 EC50 = 111 nM T37693 C6S2IH 46873203 EC50 = 0.8 nM T37693 C6NK0P 46873310 EC50 = 33 nM T37693 C02UDG 46873409 EC50 = 818 nM T37693 CW0UE4 46873411 EC50 = 2 nM T37693 CU95VF 46873412 EC50 = 3 nM T37693 CEX7G9 46873414 EC50 = 1.5 nM T37693 CFYJ67 46873415 EC50 = 0.9 nM T37693 CRU34K 46873515 EC50 = 31 nM T37693 CV8F7U 46873516 EC50 = 14 nM T37693 C4DQ0A 46880367 Ki > 1000 nM T37693 C6OE4K 46880408 Ki > 1000 nM T37693 CSE86Q 46880409 Ki = 330 nM T37693 C2A3WU 46880410 Ki = 248 nM T37693 C4GQH2 46880411 Ki = 179 nM T37693 C6X7SW 46880499 Ki > 1000 nM T37693 C9XJ0K 46880500 Ki > 1000 nM T37693 C6N8WX 46880632 Ki > 1000 nM T37693 CKH6J7 46884054 IC50 = 1000 nM T37693 CVY2T4 46888365 IC50 = 5200 nM T37693 CO7M5J 46888366 IC50 = 14000 nM T37693 CLS1G3 46888367 IC50 = 2700 nM T37693 CGD6T5 46888386 IC50 = 1900 nM T37693 C13SVO 46888387 IC50 = 1200 nM T37693 C9G2HI 46888388 IC50 = 9400 nM T37693 C5D2CK 46888389 IC50 = 56 nM T37693 CME5D6 46888413 IC50 = 17000 nM T37693 CDUM26 46888645 IC50 = 3000 nM T37693 CTN16E 46888688 IC50 = 1400 nM T37693 C4SX5W 46888719 IC50 = 1300 nM T37693 CT8E9F 46888720 IC50 = 3300 nM T37693 CP75RD 46888721 IC50 = 350 nM T37693 C9Z2CO 46888748 IC50 = 500 nM T37693 CR7HN9 46888749 IC50 = 2200 nM T37693 C06HUF 46888750 IC50 = 1400 nM T37693 CEMZ98 46888775 IC50 = 530 nM T37693 CYT7P0 46888776 IC50 = 3400 nM T37693 CJDH10 46888777 IC50 = 1400 nM T37693 CM6S8Z 46888778 IC50 = 2300 nM T37693 C7R9KO 46889225 Ki = 325 nM T37693 C9R0CB 46890855 IC50 = 6300 nM T37693 CN5E1A 46890915 IC50 > 2000 nM T37693 C6OSC8 46890967 IC50 > 2000 nM T37693 CA2V8W 46891079 IC50 = 2920 nM T37693 COQ1S6 46891146 IC50 = 3790 nM T37693 CX45SG 46896277 Ki = 19.5 nM T37693 CC96SR 46896492 Ki = 13.6 nM T37693 CFB10Q 46896493 Ki = 51.1 nM T37693 C54GCB 46896692 Ki = 9.5 nM T37693 CC9FZ0 46898063 IC50 = 549 nM T37693 CU65IN 46899610 Ki = 10000 nM T37693 CI5J2G 46899611 Ki = 25000 nM T37693 C09NDY 46899612 Ki = 20000 nM T37693 C0XJ8M 46899613 Ki = 25000 nM T37693 CL4HA6 46901905 Ki = 20000 nM T37693 CH5C9E 46901906 Ki = 25000 nM T37693 COS8Q6 46901907 Ki = 15000 nM T37693 CQ6VK0 46902047 Ki = 5000 nM T37693 CT3KO0 46902048 Ki = 8700 nM T37693 CDL21H 46902049 Ki = 35000 nM T37693 C0R7CX 46902050 Ki = 2700 nM T37693 CS42YR 46902051 Ki = 15000 nM T37693 C7T2GX 46909057 IC50 = 150000 nM T37693 CJ67QO 46909577 Ki = 1.63 nM T37693 CL47EI 46911790 Ki = 0.25 nM T37693 CD31GS 46914568 Ki = 20.6 nM T37693 CCDY16 46914722 Ki = 3881 nM T37693 C43TQI 46914723 Ki = 73.2 nM T37693 CZS28Q 46914724 Ki = 65.9 nM T37693 C1PK8H 46914725 Ki = 0.7 nM T37693 CD1T3Z 46914726 Ki = 2.3 nM T37693 CIG17Z 46914868 Ki = 4.2 nM T37693 CMV18T 46914869 Ki = 8.3 nM T37693 CXGF68 46914870 Ki = 11 nM T37693 C10IJF 46914871 Ki = 16 nM T37693 C5US1J 46915018 Ki = 44.8 nM T37693 C72YRK 46915019 Ki = 59.3 nM T37693 C48PXG 46915021 Ki = 125.7 nM T37693 C08DTP 46915022 Ki = 41.9 nM T37693 C4TXE9 46915181 Ki = 21.5 nM T37693 C3ZLI4 46915182 Ki = 52.6 nM T37693 C2HQ5I 46915183 Ki = 51 nM T37693 C5T4EW 46915184 Ki = 71.6 nM T37693 C9ZMB6 46915338 Ki = 181 nM T37693 CK36UG 46915339 Ki = 343 nM T37693 C15YSX 46915340 Ki = 8.8 nM T37693 CT1P4V 46915341 Ki = 65.4 nM T37693 CIDJ51 46915342 Ki = 0.7 nM T37693 C24CMT 46915484 Ki = 8 nM T37693 CP3T2G 46915629 Ki = 7.3 nM T37693 C3L2BF 46915632 Ki = 16.9 nM T37693 CR1K7X 46915633 Ki = 56.6 nM T37693 CN0A1F 46915770 Ki = 49.8 nM T37693 C26GKJ 46915774 Ki = 1122018.45 nM T37693 CHG94W 46915775 Ki = 59 nM T37693 C90CHW 46915915 Ki = 4.4 nM T37693 CIO5Y8 46916568 Ki = 35 nM T37693 CZ4PY1 46919791 Ki = 3.981 nM T37693 CJ70AD 46919792 Ki = 0.3981 nM T37693 CT8Z7B 48127247 Ki = 8 nM T37693 CS4LC8 48131648 Ki = 200 nM T37693 CWEH82 48134599 Ki = 53 nM T37693 CN4Q7O 49779469 EC50 = 12.2 nM T37693 CPW56Y 49780575 Ki = 1285 nM T37693 CB68TP 49780791 Ki = 496 nM T37693 C2B6NH 49780792 Ki = 451 nM T37693 CNCG41 49780793 Ki = 553 nM T37693 CO7W4M 49781019 Ki > 2500 nM T37693 C3B1WZ 49781020 Ki > 2500 nM T37693 C4OJ3P 49781021 Ki = 1037 nM T37693 CKE6A5 49781237 Ki = 683 nM T37693 CZ7M0W 49781238 Ki > 25000 nM T37693 CB91JD 49781239 Ki > 25000 nM T37693 C9I2YR 49781454 Ki > 2500 nM T37693 C1NLT8 49781455 Ki > 2500 nM T37693 CB24YU 49781456 Ki > 2500 nM T37693 CR4KL0 49781457 Ki = 622 nM T37693 CNW96U 49781458 Ki = 419 nM T37693 C2DWZ4 49781682 Ki = 305 nM T37693 CAD7R3 49781683 Ki > 25000 nM T37693 CCW7S8 49781684 Ki = 1934 nM T37693 C35OZF 49781685 Ki = 265 nM T37693 CXPZ67 49781896 Ki = 426 nM T37693 CR8X9A 49782343 Ki = 5.88 nM T37693 CFEW08 49782344 Ki = 1.62 nM T37693 C20DKN 49782345 Ki = 1.63 nM T37693 CQ98ZG 49782560 Ki = 7.02 nM T37693 C6KZL5 49782561 Ki = 3.34 nM T37693 C40DLI 49782782 Ki = 32.6 nM T37693 C9FV3Z 49782783 Ki = 15.1 nM T37693 CWA1R0 49782784 Ki = 11.9 nM T37693 CQU0W8 49783205 Ki = 1.32 nM T37693 C7D1ZA 49783408 Ki = 3.02 nM T37693 CA4T6N 49783410 Ki = 5.13 nM T37693 CL1V2G 49796909 Ki = 420 nM T37693 CM8CT6 49819854 EC50 = 7.8 nM T37693 CAP20Y 49819855 EC50 = 7.4 nM T37693 C2H3LB 49819856 EC50 = 10.9 nM T37693 CY54HV 49820008 EC50 = 5.5 nM T37693 C1XHJ3 49820009 EC50 = 3.2 nM T37693 C1I6ES 49820010 EC50 = 8.7 nM T37693 C1UBA0 49820012 EC50 = 60 nM T37693 CM93PJ 49820013 EC50 = 1.9 nM T37693 CC91QZ 49820163 EC50 = 1.9 nM T37693 C45VYH 49820164 EC50 = 23 nM T37693 CZX25W 49820165 EC50 = 26 nM T37693 CAU16J 49820166 EC50 = 22 nM T37693 CQ78GC 49820167 EC50 = 5.8 nM T37693 CI26US 49820318 Ki = 0.26 nM T37693 C5SYJ4 49820319 Ki = 15.2 nM T37693 CHI43J 49820320 Ki = 6.4 nM T37693 CS94OJ 49820321 Ki = 9.6 nM T37693 CM9E4A 49820322 Ki = 9 nM T37693 CU0P1L 49820323 Ki = 24.1 nM T37693 C3TV4W 49820467 Ki > 1000 nM T37693 CO09HC 49820468 Ki = 195.8 nM T37693 CQCN46 49820469 EC50 = 39.9 nM T37693 CXW48C 49820470 Ki > 1000 nM T37693 C9ZFO5 49820471 Ki = 189.4 nM T37693 CW9NS8 49820472 Ki > 1000 nM T37693 C1UGS6 49820621 Ki = 24.4 nM T37693 C2RVE4 49820623 Ki > 1000 nM T37693 C7ZY1V 49820624 Ki = 13.4 nM T37693 CKO61F 49820625 Ki > 1000 nM T37693 CH73VZ 49820626 EC50 = 11.9 nM T37693 C1UR2D 49820779 Ki = 36.5 nM T37693 CQ6XE4 49820780 Ki > 1000 nM T37693 C8PR2X 49820781 Ki > 1000 nM T37693 CDE3A1 49820782 Ki > 1000 nM T37693 CG9H5Z 49820783 Ki = 414 nM T37693 C0GD7O 49820784 Ki = 10.2 nM T37693 C7MR2D 49840760 EC50 = 14 nM T37693 CN89JQ 49840830 EC50 = 158 nM T37693 C6QS1A 49840831 Ki = 1.8 nM T37693 CFK8J2 49840832 Ki = 0.7 nM T37693 CM0D5J 49840833 Ki = 13.2 nM T37693 CRV02J 49840834 Ki = 91.1 nM T37693 CC05PM 49840907 EC50 = 17 nM T37693 C9JE6I 49840908 EC50 = 27 nM T37693 CXI14S 49840909 EC50 = 164 nM T37693 CR5M8V 49840911 EC50 = 25 nM T37693 C9K1PB 49847679 EC50 = 0.67 nM T37693 CZK27C 49848443 EC50 = 56 nM T37693 C32PJB 49855337 EC50 = 3.162 nM T37693 CQZB40 49861285 Ki = 26.92 nM T37693 CWJ2C0 49862666 Ki = 0.7943 nM T37693 C4Q9BH 49863941 Ki = 19 nM T37693 CC46ZO 49863942 Ki = 1300 nM T37693 CV47MH 49864283 Ki = 5 nM T37693 C9UAP2 49864284 Ki = 400 nM T37693 CKZ76J 49864285 Ki = 900 nM T37693 C7Y9FB 49864287 Ki = 2.4 nM T37693 C5ABZ0 49865134 IC50 = 1140 nM T37693 CF9C1E 49865136 IC50 = 3631 nM T37693 C0Y5ZU 49865137 IC50 = 505 nM T37693 CG98LM 49865191 IC50 = 430 nM T37693 CWG85A 49865311 IC50 = 76.8 nM T37693 CI63HS 49865364 IC50 = 265 nM T37693 CPEF69 49865365 IC50 = 124 nM T37693 CB2Y0O 49865414 IC50 = 73.6 nM T37693 C5OMV3 49865415 IC50 = 27.6 nM T37693 C7Y1GV 49865614 Ki = 79 nM T37693 CHC10N 49865615 Ki = 19.8 nM T37693 CSGK87 49865616 Ki = 26.6 nM T37693 CD0CJ2 49865617 Ki = 22.5 nM T37693 CTC3W1 49865618 Ki = 15 nM T37693 C1VUG0 49865655 Ki = 103 nM T37693 C7AWN5 49865656 Ki = 11.9 nM T37693 CN83QV 49865683 Ki = 3.4 nM T37693 C2JX4A 49865713 Ki = 9.1 nM T37693 C8Y9CP 49866230 Ki = 13.3 nM T37693 CS7TP4 49866255 Ki = 8 nM T37693 C0BQ4U 49890666 Ki > 10000 nM T37693 C2RY0J 50878551 Ki > 10000 nM T37693 CKBS87 50898695 IC50 = 1000 nM T37693 CFA38L 50898696 Ki = 1030 nM T37693 CP46YL 50898697 Ki = 2040 nM T37693 C3PIV5 50898698 Ki > 10000 nM T37693 CI2FV7 50899193 EC50 < 100 nM T37693 C3B0HL 50907287 Ki = 1496.2 nM T37693 CNM78T 50907288 Ki = 795.7 nM T37693 C7AVR3 50907289 Ki = 205.9 nM T37693 C0RGF2 50907490 Ki = 2344.4 nM T37693 CGHI15 50907491 Ki = 383.3 nM T37693 C13OJL 50907492 Ki = 255.1 nM T37693 CMT0K4 50907493 Ki = 1953.3 nM T37693 CHAB52 50907494 Ki = 459.8 nM T37693 CC0B4J 50907495 Ki = 495.3 nM T37693 C20WYJ 50907705 Ki = 3200.5 nM T37693 C9H8UP 50907706 Ki = 487.3 nM T37693 CB7V4R 50907707 Ki = 204.8 nM T37693 C7R5KQ 50907708 Ki = 365.5 nM T37693 C2X9WV 50907709 Ki = 1132.4 nM T37693 C0MZA9 50907710 Ki = 14.6 nM T37693 C6RF7I 50907920 Ki = 5.7 nM T37693 CW39DE 50907921 Ki = 52.4 nM T37693 COCB87 50907922 Ki = 237.3 nM T37693 CM7W3P 50907923 Ki = 1796.8 nM T37693 CK6MT8 50907924 Ki = 20.2 nM T37693 C1S4IB 50907925 Ki = 121.5 nM T37693 CS8MX3 50908151 Ki = 133.5 nM T37693 CT0IA2 50908152 Ki = 135.5 nM T37693 CVC8L6 50908153 Ki = 163.4 nM T37693 C1YF6I 50915132 EC50 = 3.7 nM T37693 CC0DR4 50941835 EC50 = 21 nM T37693 C9WA0L 51029725 EC50 = 2.3 nM T37693 C2IH9K 51030930 EC50 = 5.9 nM T37693 CX4PF6 51030931 EC50 = 1.2 nM T37693 CVSA07 51035170 Ki = 49.6 nM T37693 C31UWX 51042138 Ki = 0.7 nM T37693 CAO41L 51351511 EC50 = 67 nM T37693 CQ3TF0 51353567 Ki = 1.6 nM T37693 C9AZ3J 51357040 Ki = 900 nM T37693 C8T1BE 51357043 Ki = 1370 nM T37693 C3BRM2 51357044 Ki = 400 nM T37693 CIZ96K 51357316 Ki = 680 nM T37693 C5RXF2 51357319 Ki = 500 nM T37693 C6G9SM 51357595 Ki = 130 nM T37693 C1R0DP 51357597 Ki = 1800 nM T37693 CU0I5S 51357598 Ki = 7700 nM T37693 CE3H6X 51357599 Ki = 2000 nM T37693 CGV79B 51357600 Ki = 490 nM T37693 C6S1KB 51357868 Ki = 1600 nM T37693 CD9FL1 52918122 IC50 = 33 nM T37693 CRWO47 52918123 IC50 = 16 nM T37693 CC2O0K 52918124 IC50 = 7.3 nM T37693 CTF2N5 52940939 Ki = 4.4 nM T37693 C69TMB 52941604 Ki = 2500 nM T37693 C9JYF6 52941900 EC50 = 15 nM T37693 CA67NY 52941914 Ki = 265 nM T37693 CJZ5H2 52942016 Ki = 0.4 nM T37693 CS0J3G 52942068 Ki = 249 nM T37693 C8EI5P 52942075 Ki = 23 nM T37693 CN80LW 52942141 Ki = 8.4 nM T37693 CD17ZG 52942847 Ki = 71 nM T37693 CF4E2M 52942849 Ki = 171 nM T37693 CP1U7X 52943266 Ki = 258 nM T37693 C04AXC 52943267 Ki = 0.8 nM T37693 C9NI2H 52943412 Ki = 4.2 nM T37693 CG9A2Y 52943719 Ki > 10000 nM T37693 C5PRN4 52944075 Ki = 0.4 nM T37693 CE7K2D 52944154 IC50 = 3400 nM T37693 CA3G2Y 52944330 Ki = 555 nM T37693 C5B7KN 52944375 Ki > 10000 nM T37693 CJVO41 52944404 Ki = 41 nM T37693 CJC80T 52944536 Ki = 452 nM T37693 CAS17G 52944568 Ki = 0.7 nM T37693 CXTP85 52944569 Ki = 7.5 nM T37693 CL0IT3 52944886 Ki > 10000 nM T37693 C46GIZ 52944912 Ki > 10000 nM T37693 CV50BI 52945743 Ki = 1.8 nM T37693 CAIY83 52945800 Ki = 70 nM T37693 C4MXS5 52945877 Ki = 1.5 nM T37693 CUL1B5 52946095 Ki > 10000 nM T37693 C0N1WL 52946548 Ki = 1.4 nM T37693 CDR3S5 52946769 Ki = 28 nM T37693 CAG4K7 52946871 Ki = 0.35 nM T37693 CTY4D9 52946998 Ki = 3.1 nM T37693 CB2LF5 52947371 Ki > 10000 nM T37693 CQWZ29 52947376 Ki > 10000 nM T37693 C87AFQ 52947385 Ki = 2250 nM T37693 CC9Q1I 52947697 Ki > 10000 nM T37693 C5H7EL 52948053 Ki > 10000 nM T37693 CP3W7X 52948135 Ki = 790 nM T37693 CJZ97W 52948160 Ki = 2.5 nM T37693 CM03HL 52948165 Ki = 78 nM T37693 CF5UM8 52948206 Ki = 9 nM T37693 CIN5P4 52948246 Ki = 1 nM T37693 CR91MP 52948314 Ki = 16 nM T37693 CT0XY2 52948592 Ki > 10000 nM T37693 CN16UM 52948595 Ki > 10000 nM T37693 CIKX21 52949380 Ki = 8430 nM T37693 CJ9AX7 52949381 Ki = 0.9 nM T37693 CSH7T5 52949398 Ki = 0.2 nM T37693 CO9I0S 52949599 Ki = 0.5 nM T37693 C09DXM 52949805 Ki > 10000 nM T37693 C9ADM3 52950114 Ki > 10000 nM T37693 C9C1FN 52951268 Ki > 10000 nM T37693 CXF3Z8 52951269 Ki = 2180 nM T37693 C6AVI3 52951270 Ki > 10000 nM T37693 C5DRM0 52951271 Ki > 10000 nM T37693 C1LD4S 52951378 Ki > 10000 nM T37693 C8OMI5 52951379 Ki > 10000 nM T37693 CI47GU 52951380 Ki > 10000 nM T37693 CM0D9Z 52951381 Ki = 226 nM T37693 CV1BX8 52951382 Ki = 655 nM T37693 CLY37M 52951383 Ki > 10000 nM T37693 CC63FQ 52951479 Ki > 10000 nM T37693 C06YFP 52951480 Ki = 2460 nM T37693 CPA2G4 52951481 Ki = 1890 nM T37693 CYP0I3 52951482 Ki = 2750 nM T37693 CAF5K3 52951483 Ki = 234 nM T37693 CZC4B0 52951484 Ki = 2370 nM T37693 CI5M7G 52951606 Ki = 175 nM T37693 CN39RI 52951607 Ki > 10000 nM T37693 C51UGF 52951608 Ki > 10000 nM T37693 C6UQ3N 53233689 EC50 = 61 nM T37693 CJXH50 53316569 Ki > 3000 nM T37693 CWCA05 53316975 Ki = 6.5 nM T37693 C8S0EL 53317367 EC50 = 87 nM T37693 C7M9BI 53317422 EC50 = 61 nM T37693 CS8C4D 53317423 EC50 = 5 nM T37693 C9XJ4D 53317638 Ki = 9 nM T37693 CDZ2R3 53318301 Ki = 52.6 nM T37693 CT8OS9 53318302 Ki = 3.9 nM T37693 C4GL7O 53318303 Ki = 9.7 nM T37693 CW6J9C 53318654 EC50 = 10 nM T37693 C7IH8G 53318655 EC50 = 5 nM T37693 CQSZ57 53318656 EC50 = 4 nM T37693 C2DRC3 53318712 EC50 > 1000 nM T37693 CF1BS7 53318713 EC50 = 25 nM T37693 CP6X3G 53318779 EC50 = 11 nM T37693 C2SY3X 53318780 EC50 = 70 nM T37693 CHC3R5 53319210 EC50 = 6.5 nM T37693 CJ0M5I 53319626 Ki = 8 nM T37693 C6V5OU 53319661 Ki = 25.5 nM T37693 C8R6XB 53319972 EC50 = 8 nM T37693 CW8EQ3 53320023 EC50 = 8 nM T37693 CRS79K 53320272 EC50 = 113 nM T37693 CI80DM 53320925 Ki = 16 nM T37693 C4VAP1 53321340 EC50 = 218 nM T37693 CJE6F1 53322251 Ki = 3 nM T37693 CBD23U 53322256 Ki = 2.4 nM T37693 CFQY21 53322288 Ki = 3.5 nM T37693 CZA30O 53322289 Ki = 1.2 nM T37693 CVP47L 53322598 EC50 = 3 nM T37693 C8JLS1 53322599 EC50 = 130 nM T37693 CY9ZK2 53322600 EC50 = 510 nM T37693 C1UJ5C 53322647 EC50 = 169 nM T37693 CQP16M 53322648 EC50 = 16 nM T37693 CTZ0Q9 53323192 EC50 = 25 nM T37693 CO7ED9 53323994 EC50 = 9 nM T37693 CNJQ28 53323995 EC50 = 6 nM T37693 CP8CN3 53323996 EC50 = 9 nM T37693 CS9I8F 53323997 EC50 = 5 nM T37693 CNMF87 53324282 EC50 = 10 nM T37693 CO7BF5 53324934 Ki = 5.7 nM T37693 CN6VT3 53324935 Ki = 2.7 nM T37693 CQ7ME2 53325220 EC50 = 4 nM T37693 CF2DQ0 53325221 EC50 = 24 nM T37693 C6T9OP 53325289 EC50 > 1000 nM T37693 CFCT05 53325377 EC50 = 14 nM T37693 C2VR6O 53326220 Ki = 10 nM T37693 CW7PM5 53326510 EC50 = 5 nM T37693 C1ZF7K 53326560 EC50 = 412 nM T37693 C7NB8Z 53326561 EC50 > 1000 nM T37693 C8HB2L 53341132 EC50 < 100 nM T37693 CK3I2Y 53353783 Ki = 42 nM T37693 C85YKL 53357396 EC50 < 100 nM T37693 CYG6Q1 53358318 EC50 = 2.7 nM T37693 CKCW59 53358319 EC50 = 11 nM T37693 C9XKB7 53358426 EC50 = 5.3 nM T37693 C5ZHE4 53377393 Ki > 10000 nM T37693 C3X7OW 53386375 EC50 = 22.4 nM T37693 CW91SC 53387189 Ki = 0.6 nM T37693 CKSB51 53387350 Ki = 8.5 nM T37693 CKE02W 53387351 Ki = 0.2 nM T37693 CH37DN 53387419 Ki > 2000 nM T37693 CFJG62 53387420 Ki > 2000 nM T37693 C7HRK8 53387421 Ki > 2000 nM T37693 CQZF69 53387584 Ki > 2000 nM T37693 CM47GI 53387585 Ki > 2000 nM T37693 CQ81LN 53387586 Ki = 379 nM T37693 CN67QX 53387587 Ki = 450 nM T37693 C0GI9B 53387746 Ki = 84.9 nM T37693 CS8B2H 53392078 Ki = 6.9 nM T37693 C6RKL5 53392169 Ki = 220 nM T37693 CM8T0J 53392248 Ki = 1 nM T37693 CGZD15 53392250 Ki = 22.9 nM T37693 CZ18IO 53392334 Ki = 430 nM T37693 CE29LJ 53392335 Ki = 1180 nM T37693 CLBE83 53392336 Ki = 133 nM T37693 CQ95FH 53392951 Ki > 10000 nM T37693 C82NLO 53394455 Ki = 78.3 nM T37693 CV5NQ4 53476894 EC50 = 22.4 nM T37693 C6VLZ9 53483967 Ki = 900 nM T37693 CUBX46 53483982 Ki = 1790 nM T37693 CI91KL 53484076 Ki = 253 nM T37693 CM5AI6 53484092 Ki = 1160 nM T37693 C2TP3Z 53494923 Ki = 2.8 nM T37693 CP8MN1 53494924 Ki = 22 nM T37693 CG9L7V 53494925 Ki = 0.7998 nM T37693 CO1K2X 53494926 Ki = 1.4 nM T37693 CP6A8N 53749463 Ki = 1.9 nM T37693 CG9QN4 54208075 Ki = 72.95 nM T37693 C0D8TA 54213246 Ki = 17.99 nM T37693 CR4N3X 54577602 Ki = 7.5 nM T37693 CX91HL 54579950 EC50 > 20000 nM T37693 C7I3ZC 54579951 EC50 = 2865 nM T37693 CDO2B0 54580174 IC50 = 44 nM T37693 CS2PI0 54580175 IC50 = 21 nM T37693 C5N2YX 54580194 IC50 = 0.55 nM T37693 C5AVO4 54580197 IC50 = 41 nM T37693 CZG6L5 54580223 IC50 = 5.9 nM T37693 C40PMJ 54580224 IC50 = 155 nM T37693 CJ7NC5 54580225 IC50 = 493 nM T37693 C1M4UV 54580226 IC50 = 338 nM T37693 CB37OP 54580227 IC50 = 5.5 nM T37693 CVU32Y 54580228 IC50 = 1.4 nM T37693 CFE51I 54580229 IC50 = 6.1 nM T37693 C4VGN2 54580230 IC50 = 135 nM T37693 C9G0UX 54580231 IC50 = 30 nM T37693 CKLR94 54580466 EC50 = 450 nM T37693 CSR9V2 54580931 EC50 = 8.4 nM T37693 C9YD6K 54581168 IC50 = 21 nM T37693 C72HZB 54581169 IC50 = 69 nM T37693 C43FAB 54581198 IC50 = 1286 nM T37693 C9FO1C 54581199 IC50 = 0.82 nM T37693 C4P8NW 54581223 IC50 = 0.53 nM T37693 C4AE7R 54581224 IC50 = 11 nM T37693 CUC36A 54581225 IC50 = 395 nM T37693 CVK59Q 54581226 IC50 = 41 nM T37693 C7ZL8M 54581476 EC50 = 1940 nM T37693 C8K7RL 54581988 EC50 = 13150 nM T37693 C6FU2I 54581989 EC50 = 1350 nM T37693 CF39HJ 54582173 IC50 = 0.3 nM T37693 C3T7CY 54582249 IC50 = 21 nM T37693 C67TLK 54582250 IC50 = 106 nM T37693 CJX1K9 54582251 IC50 = 35 nM T37693 C3GM8O 54582252 IC50 = 4 nM T37693 CP64NQ 54582479 EC50 = 168 nM T37693 C5PZ4A 54582480 EC50 = 2.7 nM T37693 CG3FA5 54582481 EC50 = 1700 nM T37693 CFG5J2 54582482 EC50 = 14850 nM T37693 C61IJU 54582925 EC50 = 750 nM T37693 CJ0F2K 54583160 IC50 = 139 nM T37693 C08ONK 54583196 IC50 = 22 nM T37693 CCS50N 54583230 IC50 = 30 nM T37693 C0ET3G 54583455 EC50 > 20000 nM T37693 CD2BN6 54583456 EC50 > 20000 nM T37693 CDF83A 54583457 EC50 = 150 nM T37693 C4G9CW 54583926 EC50 = 2300 nM T37693 C06IDY 54583927 EC50 = 814 nM T37693 CNQC76 54584153 IC50 = 7 nM T37693 CJZS79 54584190 IC50 = 3.38 nM T37693 C0K9SP 54584191 IC50 = 6.3 nM T37693 CX2EJ4 54584192 IC50 = 124 nM T37693 C8THZ7 54584193 IC50 = 16 nM T37693 CXZL01 54584423 EC50 > 20000 nM T37693 CNVG29 54584424 EC50 = 215 nM T37693 CFJ1G3 54584425 EC50 = 26 nM T37693 C37TZQ 54584868 EC50 = 135 nM T37693 C4EB1D 54585060 IC50 = 0.7 nM T37693 COQ86B 54585087 IC50 = 1.7 nM T37693 CVG86Q 54585088 IC50 = 3 nM T37693 CA7ZM4 54585089 IC50 = 92 nM T37693 CV6PE4 54585090 IC50 = 36 nM T37693 C0B6DK 54585147 IC50 = 0.62 nM T37693 CK9N2B 54585148 IC50 = 12 nM T37693 C47CQF 54585149 IC50 = 12 nM T37693 C7TF3G 54585381 EC50 = 85 nM T37693 C19LYO 54585382 EC50 = 96 nM T37693 C3CIW8 54585835 EC50 = 2045 nM T37693 C60ZBV 54585836 EC50 = 4030 nM T37693 CUI9N5 54585837 EC50 = 177 nM T37693 CS5V9Y 54586103 IC50 = 938 nM T37693 CJLB09 54586104 IC50 = 2175 nM T37693 CY7XN2 54586105 IC50 = 1.6 nM T37693 C78MRT 54586106 IC50 = 29 nM T37693 CQ74VR 54586107 IC50 = 156 nM T37693 CYCN52 54586108 IC50 = 3471 nM T37693 CE7WF1 54586109 IC50 = 193 nM T37693 CNHM97 54586338 EC50 > 20000 nM T37693 CM14QB 54586803 EC50 = 1690 nM T37693 CG56XR 54586804 EC50 = 157 nM T37693 CQWI92 54586805 EC50 = 107 nM T37693 C4L5SW 54586806 EC50 = 426 nM T37693 CMF92B 54587073 IC50 = 24 nM T37693 CM6Q8R 54587074 IC50 > 17000 nM T37693 CK6Q9F 54587075 IC50 = 0.14 nM T37693 CO4R1F 54587104 IC50 = 358 nM T37693 C0RU3W 54587105 IC50 = 1045 nM T37693 C1L3SH 54587106 IC50 = 810 nM T37693 C3AR4O 54587107 IC50 = 1357 nM T37693 CA37WI 54587108 IC50 = 282 nM T37693 CZ23AJ 54587109 IC50 = 56 nM T37693 CT8GH6 54587110 IC50 = 62 nM T37693 CBI84E 54587111 IC50 = 140 nM T37693 CCOF62 54587112 IC50 = 26 nM T37693 C4XT9S 54587370 EC50 = 20 nM T37693 C4GJ1Z 54587371 EC50 = 87 nM T37693 CB49IH 54587372 EC50 = 49 nM T37693 C1Q5RX 54587373 EC50 = 111 nM T37693 C6H9US 54592384 Ki = 2.5 nM T37693 CUV69N 54669855 Ki = 180 nM T37693 CU9W8M 54680181 Ki > 1000 nM T37693 C2DWJ5 54683138 EC50 = 2.4 nM T37693 CDR58P 54732041 Ki = 29.4 nM T37693 CJON78 54732042 Ki = 15 nM T37693 CE61UL 54752945 EC50 = 7.943 nM T37693 CW28JF 54752946 Ki = 50.12 nM T37693 C3P9HQ 54752947 Ki = 25.12 nM T37693 CG16QF 54769828 Ki = 1380.38 nM T37693 C8G2CW 54769829 Ki = 10.2 nM T37693 CU09YW 54769830 Ki = 1580 nM T37693 C8IH2D 56597771 IC50 > 10000 nM T37693 CQ69YX 56599474 IC50 > 10000 nM T37693 CX8BT4 56642292 Ki = 39.81 nM T37693 C23NFV 56642293 Ki = 63.1 nM T37693 CU9D7V 56642294 Ki = 7.943 nM T37693 C9X8UN 56642295 Ki > 1000 nM T37693 C26KYO 56642422 Ki > 1000 nM T37693 C8SXT3 56642423 Ki = 630.96 nM T37693 C0A5ML 56642424 Ki = 630.96 nM T37693 C3AC0D 56642425 EC50 = 6.31 nM T37693 CD8EG3 56642426 Ki = 316.23 nM T37693 CW4V3C 56642427 Ki = 199.53 nM T37693 CZ7O2R 56642428 Ki = 501.19 nM T37693 CE2B6T 56642541 Ki = 50.12 nM T37693 C51HFJ 56650338 Ki = 3594 nM T37693 CV54JA 56650343 Ki = 84.5 nM T37693 C3NZE8 56650679 Ki = 35.4 nM T37693 C40NSU 56650681 Ki = 1609 nM T37693 C80VOR 56650683 Ki = 51.8 nM T37693 CBG07N 56651017 Ki = 288.5 nM T37693 C5LXO6 56651352 Ki = 225 nM T37693 C8BCD3 56651353 Ki = 403 nM T37693 CDI6S9 56651354 Ki = 83 nM T37693 C4U5MS 56651355 Ki = 208 nM T37693 CWX71K 56651356 Ki = 101 nM T37693 C6BN9F 56651357 Ki = 20 nM T37693 CSG5C1 56651358 Ki = 600 nM T37693 C3L7DS 56651692 Ki = 91 nM T37693 CY8PJ2 56651694 Ki = 215 nM T37693 CUJQ83 56651696 Ki = 1367 nM T37693 CWD2M5 56651697 Ki = 26.5 nM T37693 CQ6A1S 56651698 Ki = 35.3 nM T37693 C60STN 56652049 Ki = 171.1 nM T37693 CS6MJ7 56658151 Ki = 4010 nM T37693 C3WAG8 56659407 EC50 = 0.43 nM T37693 C9IU7P 56659423 EC50 = 51 nM T37693 CFN58G 56659453 Ki > 10000 nM T37693 C25NUZ 56659454 Ki > 10000 nM T37693 C8F2LW 56661658 Ki = 4520 nM T37693 CKLR96 56661659 Ki = 2270 nM T37693 CI2E6F 56661776 Ki = 1010 nM T37693 C5B2WH 56662770 Ki = 486 nM T37693 CWS52M 56662852 EC50 = 12 nM T37693 CV08JQ 56662872 EC50 = 39 nM T37693 CPSB19 56662902 Ki > 10000 nM T37693 CZXH42 56666243 Ki > 10000 nM T37693 CHB2S8 56666353 EC50 = 425 nM T37693 C0J2LE 56666384 Ki > 10000 nM T37693 CV10RX 56668301 Ki = 3290 nM T37693 CNWQ23 56668510 Ki = 60 nM T37693 CA3ZL8 56668680 Ki = 780 nM T37693 CRV05W 56669650 Ki = 23 nM T37693 CAX2K8 56669651 Ki = 0.043 nM T37693 CZ62XE 56669764 EC50 = 32 nM T37693 CP8BD9 56669765 EC50 = 1.2 nM T37693 CU63SK 56669766 EC50 = 6.5 nM T37693 C4P8XI 56669767 EC50 = 132 nM T37693 C8L9GU 56669768 EC50 = 82 nM T37693 CL10NC 56669769 EC50 = 25 nM T37693 C7PBS6 56669770 EC50 = 106 nM T37693 C6R9VZ 56669796 Ki > 10000 nM T37693 CHLT70 56669797 Ki > 10000 nM T37693 CA3V1W 56673163 Ki = 2400 nM T37693 C5MF0W 56673243 EC50 = 8 nM T37693 C7WZQ1 56673258 EC50 = 67 nM T37693 C7SE6V 56673308 Ki > 10000 nM T37693 CK64EV 56675389 Ki = 3443 nM T37693 C17MNC 56676487 Ki > 10000 nM T37693 CWY8S6 56676569 EC50 = 5 nM T37693 C8V4YQ 56676584 EC50 = 199 nM T37693 C8D5KV 56676585 EC50 = 9.6 nM T37693 CG8NS6 56676603 EC50 > 20000 nM T37693 C8L9MT 56676610 Ki > 10000 nM T37693 CBM0X1 56679803 Ki = 57.94 nM T37693 C2WUA5 56679804 Ki = 0.014 nM T37693 C7V8DA 56679805 Ki = 0.036 nM T37693 CUQ0K8 56679890 Ki = 260 nM T37693 C03JXE 56679953 Ki > 10000 nM T37693 CD8Z3A 56681835 Ki = 1805 nM T37693 CLQ0O1 56683134 Ki = 619.44 nM T37693 C9YJ1K 56683149 Ki = 1.023 nM T37693 CZ71FA 56683269 EC50 > 20000 nM T37693 C4PWO8 56683270 EC50 > 20000 nM T37693 C2MFV5 56835155 EC50 = 8.2 nM T37693 CP4WL5 56835156 EC50 = 7.7 nM T37693 C78GIO 56835165 Ki = 790 nM T37693 CWE8D9 56837837 Ki = 376.4 nM T37693 C6B1MZ 56837838 Ki = 0.51 nM T37693 CBXJ07 56925623 Ki = 7870 nM T37693 C8GR5O 56925624 Ki = 870 nM T37693 C1MIN3 56925625 Ki = 7870 nM T37693 C3N9CZ 56925626 Ki = 7870 nM T37693 C6VP7T 56925628 Ki = 790 nM T37693 C1HO6A 56925747 Ki = 800 nM T37693 CUB7Q2 56925748 Ki = 910 nM T37693 CHQJ12 56925749 Ki = 1160 nM T37693 C7LH9I 56925750 Ki > 10000 nM T37693 CDEM08 56925751 Ki > 10000 nM T37693 CF7QC3 56925752 Ki = 1130 nM T37693 C47TIH 56925753 Ki = 2390 nM T37693 C6X4BI 56925870 Ki = 190 nM T37693 CPS34F 56925871 Ki = 110 nM T37693 CQAD90 56925872 Ki = 380 nM T37693 C9DS8J 56925873 Ki = 1670 nM T37693 C25PRG 56925874 Ki = 7910 nM T37693 CJ3XS5 56925875 Ki = 10440 nM T37693 COM7T4 56925978 Ki = 310 nM T37693 C9IQJ4 56930623 Ki = 242.4 nM T37693 CG6E3T 56930624 Ki = 226.8 nM T37693 CEU17F 56930925 Ki = 98.5 nM T37693 CZ1NX6 56931060 Ki = 18.3 nM T37693 CP28UN 56931061 Ki = 135.2 nM T37693 CO6E0R 56931062 Ki = 19.1 nM T37693 CH36LK 56931063 Ki = 72.9 nM T37693 CH0ZA7 56931064 Ki = 454.6 nM T37693 CB6TF2 56931065 Ki = 15.8 nM T37693 CR72TI 56931190 Ki = 56.1 nM T37693 C4Q0HK 56931191 Ki = 753.8 nM T37693 C0I6QB 56931192 Ki > 10000 nM T37693 CN6J2L 56931193 Ki = 409.6 nM T37693 C9OI6H 56931194 Ki = 53.9 nM T37693 CJ86AH 56931195 Ki = 0.9 nM T37693 C08RFS 56931309 Ki = 161.7 nM T37693 CN19LG 56931310 Ki = 1.3 nM T37693 C8AGO4 56931311 Ki = 29.6 nM T37693 CD7T1G 56931312 Ki = 113.7 nM T37693 CR71AS 56931313 Ki = 1.7 nM T37693 CAM7P0 56951321 Ki = 5400 nM T37693 CW2F4U 57329634 EC50 = 490 nM T37693 C2HZB0 57341135 Ki = 4350 nM T37693 C7C2AQ 57341136 Ki = 10893 nM T37693 CPJ3F8 57341327 Ki = 7795 nM T37693 C8S4VX 57341330 Ki = 5420 nM T37693 C50JMF 57341331 Ki = 6720 nM T37693 C4CI3V 57341512 Ki = 1248 nM T37693 CJ9FN2 57341514 Ki = 4135 nM T37693 C26YHM 57341678 Ki = 3090 nM T37693 CIC4R1 57341679 Ki = 3031 nM T37693 C6WLP1 57341681 Ki = 2507 nM T37693 CVK8R4 57342713 Ki = 5504 nM T37693 CGU32A 57342714 Ki = 2217 nM T37693 CC8T6P 57342881 Ki = 2110 nM T37693 CX1Q5W 57342882 Ki = 1127 nM T37693 CX3KY7 57342883 Ki = 214 nM T37693 C4E5IK 57342884 Ki = 41 nM T37693 C6NF1A 57342885 Ki = 20000 nM T37693 CTB1X5 57343047 Ki = 17126 nM T37693 CC6T0U 57343049 Ki = 20000 nM T37693 CHQU04 57343050 Ki = 16289 nM T37693 C6AS5E 57343221 Ki = 2414 nM T37693 C5DT6K 57343222 Ki = 4914 nM T37693 CHD82G 57343223 Ki = 182 nM T37693 C7QWP1 57343224 Ki = 293 nM T37693 C3QHI6 57343388 Ki = 20000 nM T37693 CYE41Z 57343389 Ki = 2760 nM T37693 CEL9T2 57343390 Ki = 2510 nM T37693 CI5EO4 57343392 Ki = 2236 nM T37693 C4EXK2 57343552 Ki = 3349 nM T37693 C4TGD8 57343554 Ki = 5693 nM T37693 CVR4L9 57343718 Ki = 9791 nM T37693 C4JD1Z 57343719 Ki = 8459 nM T37693 C80TPF 57343720 Ki = 8721 nM T37693 CP5Q3T 57343721 Ki = 2997 nM T37693 CE6RP0 57345610 Ki = 6.6 nM T37693 C21ZIX 57345611 Ki = 20 nM T37693 C7HU4M 57345612 Ki = 13 nM T37693 C5K7QN 57387465 IC50 = 15 nM T37693 CEP0O6 57390497 Ki = 4820 nM T37693 CIV2U0 57390698 EC50 = 19 nM T37693 CSV86Y 57390762 EC50 = 4.6 nM T37693 CRFH16 57390958 Ki = 0.56 nM T37693 CG74WV 57392498 EC50 = 0.8 nM T37693 C4M2DZ 57392499 EC50 = 0.5 nM T37693 CLD7W5 57392500 EC50 = 240 nM T37693 C8X5TH 57393210 Ki = 1800 nM T37693 CZF5C6 57394209 EC50 = 1.3 nM T37693 CKW7S4 57396050 EC50 = 28 nM T37693 CM5DG7 57396051 EC50 = 26 nM T37693 CJT6Q5 57396515 Ki = 490 nM T37693 CI30KJ 57396516 Ki = 4021 nM T37693 CV3I7P 57397849 EC50 = 8.4 nM T37693 C7HOF1 57399434 EC50 = 1.2 nM T37693 CR0XE3 57399435 EC50 = 1.4 nM T37693 CP6D2M 57399436 EC50 = 23 nM T37693 C25STE 57399512 EC50 = 8.4 nM T37693 C9JLX0 57399513 EC50 = 3 nM T37693 CPU9O6 57401192 EC50 = 5.6 nM T37693 C8SW2Q 57401265 EC50 = 17 nM T37693 C75DTX 57401266 EC50 = 2.2 nM T37693 CS4YZ9 57402953 EC50 = 1.1 nM T37693 C80XAI 57403011 EC50 = 23 nM T37693 CD2YM3 57403012 EC50 = 145 nM T37693 C0BVA6 57403652 Ki = 1800 nM T37693 CH24BN 57404063 EC50 = 92 nM T37693 C3P1IN 57404070 EC50 = 29 nM T37693 CY3O0M 57441073 Ki = 0.871 nM T37693 CKOW75 57458928 Ki = 2.8 nM T37693 CP0BN7 57458937 Ki = 5.4 nM T37693 C41WFI 57507910 EC50 = 4.5 nM T37693 CIMZ13 57507911 EC50 = 6.9 nM T37693 CD7KI5 57555816 Ki = 19.95 nM T37693 C7D1JL 57606048 Ki = 15.5 nM T37693 CO2CH9 57708174 EC50 = 0.15 nM T37693 CLD68M 57780750 IC50 = 110 nM T37693 C4FNG6 57780757 IC50 = 100 nM T37693 CT12KZ 58459056 EC50 = 5.9 nM T37693 CL85HS 58459075 EC50 = 12.5 nM T37693 C35EYG 58459090 EC50 = 5 nM T37693 CV5O8N 58459093 EC50 = 6.8 nM T37693 C20RBA 58459095 EC50 = 8.1 nM T37693 C7AZ0L 58459098 EC50 = 4.3 nM T37693 C06UDC 58459099 EC50 = 4.7 nM T37693 CRNS43 58513574 EC50 = 8.9 nM T37693 CCO8I6 58513582 EC50 = 278 nM T37693 CQ52IW 58513592 EC50 = 104 nM T37693 CM7UX9 58513605 EC50 = 62 nM T37693 CRX0O9 58513615 EC50 = 4.8 nM T37693 CO9VG5 58563756 EC50 = 108 nM T37693 CQU7K0 58563758 EC50 = 0.2 nM T37693 CE4D3P 58563847 EC50 = 63 nM T37693 CSTP80 58563862 EC50 = 69 nM T37693 C9C5WJ 58682997 Ki = 32 nM T37693 CGZ72Q 58882471 EC50 = 5590 nM T37693 C50VGR 58882571 EC50 = 12 nM T37693 CEF5R0 58973328 IC50 > 10000 nM T37693 CV6R3G 58973346 IC50 = 190 nM T37693 CKC13R 58973398 IC50 = 19 nM T37693 C6ZQ3C 58973420 IC50 = 1200 nM T37693 C1WZ9B 58999139 IC50 > 5000 nM T37693 CH0C3G 59169713 Ki = 0.15 nM T37693 CYNH83 59268968 Ki > 5000 nM T37693 C4YHN9 59450165 Ki = 325 nM T37693 CH2N8X 59450184 Ki = 24 nM T37693 C8OW3Y 59450186 Ki = 13.3 nM T37693 C7JL9W 59450189 Ki = 31.8 nM T37693 C0K2HL 59699565 Ki = 79 nM T37693 CWX31A 59718742 Ki = 349 nM T37693 CA3X1B 59718743 Ki = 3 nM T37693 CQ90HR 59718804 IC50 = 2.5 nM T37693 CNK4O7 59718824 Ki = 177 nM T37693 CS4N1M 59718841 Ki = 7.3 nM T37693 CRFL45 59718847 IC50 = 1.4 nM T37693 CPAJ14 59718848 Ki = 2.8 nM T37693 CS0W6L 59718873 Ki = 0.6 nM T37693 CG7WN9 59799318 EC50 = 0.56 nM T37693 C50WFM 60005384 Ki = 101 nM T37693 CL5W4C 60145369 Ki = 16 nM T37693 CJ4I7K 60145370 Ki = 2.9 nM T37693 CLZ36M 60145371 Ki = 9 nM T37693 CP7H3F 60145372 Ki = 2 nM T37693 CST6V2 60145373 Ki = 130 nM T37693 CYER47 60145524 Ki = 2.4 nM T37693 CT32WR 60145526 Ki = 1.8 nM T37693 C94VJI 60145527 Ki = 20 nM T37693 CAKN82 60145528 Ki = 7900 nM T37693 CK54GR 60145662 EC50 = 6.31 nM T37693 CICU98 60145663 Ki = 790 nM T37693 C32PWF 60145664 Ki = 916 nM T37693 CT8ED4 60145665 Ki = 250 nM T37693 CM3C5S 60145666 Ki = 25 nM T37693 CE5J4O 60149000 EC50 = 8.8 nM T37693 CR9M5O 60150688 Ki = 1.2 nM T37693 CJ6VL2 60150697 Ki > 30000 nM T37693 C2W9BH 60150698 Ki = 59000 nM T37693 CORL92 60154838 Ki = 70.8 nM T37693 C91ITY 60154841 Ki = 377 nM T37693 CDF8J3 60154924 Ki = 50 nM T37693 C9O4VR 60154925 Ki = 110 nM T37693 CR8H4E 60154926 Ki = 98 nM T37693 CT3ZU0 60154927 Ki = 67 nM T37693 C0PME3 60154928 Ki = 11.8 nM T37693 C1G5UC 60155009 Ki = 50 nM T37693 CP6DH5 60155010 Ki = 20.5 nM T37693 CK56XU 60155011 Ki = 17.8 nM T37693 C0Q7MN 60155012 Ki = 70 nM T37693 CN8W3E 60155013 Ki = 189 nM T37693 CRY3M4 60155101 Ki = 0.37 nM T37693 CX72BW 60155102 Ki = 12.7 nM T37693 C9MGL1 60155103 Ki = 10.3 nM T37693 CD5W7S 60155104 Ki = 25.4 nM T37693 C5I9SG 60155105 Ki = 11.2 nM T37693 C1LEX2 60155185 Ki = 1.82 nM T37693 CGBH93 60155186 Ki = 22.2 nM T37693 C6TP9E 60155187 Ki = 5.73 nM T37693 CBC50Z 60155188 Ki = 11.6 nM T37693 CM81VH 60155189 Ki = 2.48 nM T37693 COYK60 60155275 Ki = 6.37 nM T37693 CL3HG6 60155276 Ki = 3.52 nM T37693 CVA6Z1 60155280 Ki = 1090 nM T37693 CR70DY 60155369 Ki = 170 nM T37693 C3F4XM 60155736 EC50 = 130 nM T37693 C27XCO 60155737 IC50 > 10000 nM T37693 CEU78G 60155738 IC50 = 5570 nM T37693 CU3H4T 60155817 EC50 > 10000 nM T37693 CQ0D2Z 60155818 IC50 = 6970 nM T37693 CV6Y9Q 60155819 IC50 > 10000 nM T37693 CVZ0D5 60155820 IC50 > 10000 nM T37693 C1TRU8 60155821 IC50 = 9130 nM T37693 CWP04U 60155822 IC50 > 10000 nM T37693 C9RH8P 60155823 IC50 > 10000 nM T37693 C2LXE9 60155915 IC50 > 10000 nM T37693 C0X6TB 60155916 IC50 > 10000 nM T37693 C18GHZ 60155917 IC50 > 10000 nM T37693 CHO64N 60155918 IC50 > 10000 nM T37693 C75SZK 60155919 EC50 > 10000 nM T37693 CD8S3V 60155920 IC50 = 8970 nM T37693 CQFG39 60155921 IC50 > 10000 nM T37693 CUY1D2 60156024 IC50 > 10000 nM T37693 CACY36 60156025 IC50 > 10000 nM T37693 CF4T0W 60156026 IC50 > 10000 nM T37693 C5PFT2 60156027 IC50 > 10000 nM T37693 C1D0WM 60168356 EC50 = 105 nM T37693 CUP40N 60168357 EC50 = 26 nM T37693 CZPG14 60168437 EC50 = 59 nM T37693 CWER04 60168627 EC50 = 46 nM T37693 CY52RD 60194851 Ki = 24 nM T37693 C1IQ4D 60194852 Ki = 188 nM T37693 C0J9IC 60194853 Ki = 47 nM T37693 CNE0W5 60194854 Ki = 78 nM T37693 CD5FM4 60194855 Ki = 4.12 nM T37693 CC0YJ5 60194856 Ki = 187 nM T37693 C9IPS3 60194934 Ki = 4.93 nM T37693 C2QP1O 60194935 Ki = 88 nM T37693 C94RWT 60194936 Ki = 1.24 nM T37693 C76HOR 60194937 Ki = 16.2 nM T37693 CPC37E 60194939 Ki = 42 nM T37693 CKE71C 60195491 Ki = 98 nM T37693 CK4JA9 60195572 Ki = 2.52 nM T37693 CP0E6D 60195573 Ki = 0.81 nM T37693 CO0P4A 60195574 Ki = 14.2 nM T37693 CVX21O 60195576 Ki = 536 nM T37693 CSL35V 60195655 Ki = 332 nM T37693 CP1AR4 60195656 Ki > 10000 nM T37693 C4H7CW 60195657 Ki = 468 nM T37693 CFNO62 60195658 Ki = 412 nM T37693 CQSK90 60195659 Ki = 18.4 nM T37693 CKB79Q 60195740 IC50 = 472 nM T37693 CAP71F 60195741 Ki = 60 nM T37693 CH84CF 60195742 Ki = 38 nM T37693 C2DPQ3 60195743 Ki = 47 nM T37693 COAS29 60195744 Ki = 22 nM T37693 C14UMZ 60195745 Ki = 9.24 nM T37693 C5M9SZ 60195831 Ki = 13.2 nM T37693 CYHG21 60195832 Ki = 15.8 nM T37693 C9VD5Y 60195833 Ki = 152 nM T37693 CWXZ73 60195835 Ki = 85 nM T37693 C8K4BZ 60195836 Ki = 0.32 nM T37693 C74ZPK 60195919 Ki = 2.34 nM T37693 C3FV2S 60195921 Ki = 38 nM T37693 CV7R1C 60195922 Ki = 10.4 nM T37693 CSD9O4 60195923 Ki = 15.3 nM T37693 C5R8ZK 60195924 Ki = 3.12 nM T37693 CP4E9Y 60196006 Ki = 8.92 nM T37693 CT0JX4 60196007 Ki = 3.74 nM T37693 C4XG7M 60196008 Ki = 56 nM T37693 CC7XE8 60196009 Ki = 7.34 nM T37693 CUW84T 60196010 Ki = 33 nM T37693 C2SU6Z 60196093 Ki = 6.78 nM T37693 CXZR09 60196094 Ki = 8.12 nM T37693 C5BVR2 60196095 Ki = 9.24 nM T37693 C2TQ6D 60196096 Ki = 3.72 nM T37693 CA7MG4 62705820 EC50 = 4.6 nM T37693 C09XDB 62705987 EC50 = 4.1 nM T37693 CL92XI 62705988 EC50 = 47.5 nM T37693 C8W6PJ 62705989 EC50 = 62 nM T37693 CUE8H3 64428131 Ki = 1000 nM T37693 CVI57W 66552190 Ki = 209.4 nM T37693 C7QR0D 66552191 Ki = 118.2 nM T37693 C98AGZ 66552193 Ki = 1551 nM T37693 C2U6BJ 66552194 Ki = 113.1 nM T37693 CVG21C 66552243 Ki = 124.8 nM T37693 C49YAZ 66552244 Ki > 1000 nM T37693 C4D9MW 66552246 Ki > 1000 nM T37693 CRW0S3 66552247 Ki > 1000 nM T37693 CL49KR 66552248 Ki > 1000 nM T37693 CVO3R5 66552305 Ki = 37.3 nM T37693 CG6L1R 66552306 Ki = 158.6 nM T37693 C8M5VA 66552307 Ki = 3006 nM T37693 CDY0W4 66552918 Ki = 587 nM T37693 CR8V2Y 66553217 IC50 > 1000 nM T37693 CUA9G5 66643149 EC50 = 0.47 nM T37693 CTS7P8 67012376 Ki > 10000 nM T37693 CKZO03 67425523 EC50 = 11.9 nM T37693 C8YE5J 67425691 EC50 = 15.9 nM T37693 CVZP79 67427023 EC50 = 106 nM T37693 CLS9K6 67433936 EC50 = 4.7 nM T37693 C9YZR3 67434101 EC50 = 8.1 nM T37693 C0LGO7 67434539 EC50 = 10.4 nM T37693 C09VFU 67434704 EC50 = 6.8 nM T37693 CL8QT1 67435171 Ki = 5.3 nM T37693 CML5F8 67450266 EC50 = 20.3 nM T37693 C8Q9MN 67455563 EC50 = 0.21 nM T37693 CT1E8P 67457326 EC50 = 2200 nM T37693 CD40IL 67458256 EC50 = 4000 nM T37693 CXQ85N 67505405 Ki > 10000 nM T37693 C6W1UQ 67519772 IC50 = 9 nM T37693 C9KZ7X 67520157 Ki = 116 nM T37693 CX1AL0 67520222 Ki = 6.699 nM T37693 C4H6ZJ 67520284 Ki = 2823 nM T37693 CX3Z9O 67953246 EC50 = 14 nM T37693 CPB54A 67953263 EC50 = 17 nM T37693 CI13QS 67953265 EC50 = 7 nM T37693 CZP98A 67953277 EC50 = 4.7 nM T37693 CE94JQ 67953283 EC50 = 0.19 nM T37693 C3T6JM 67953286 EC50 = 33 nM T37693 C06ADK 67953287 EC50 = 0.29 nM T37693 CR9BV5 67953290 EC50 = 50 nM T37693 CBK74Z 67953291 EC50 = 390 nM T37693 C19YPW 67953294 EC50 = 2.4 nM T37693 C2D6XA 67953297 EC50 = 1.1 nM T37693 CX3E4U 67953298 EC50 = 2.8 nM T37693 C42TIW 67953300 EC50 = 7.7 nM T37693 C5JUY1 67953301 EC50 = 19 nM T37693 CXI91V 67953302 EC50 = 4.2 nM T37693 CMYD72 67953303 EC50 = 0.2 nM T37693 C0I5FH 67953329 EC50 = 700 nM T37693 CT43SM 67953330 EC50 = 1.4 nM T37693 CUB95N 67953333 EC50 = 170 nM T37693 CH7FG3 67953351 EC50 = 59 nM T37693 C3YQN6 67953380 EC50 = 100 nM T37693 C0DP2O 67953418 EC50 = 38 nM T37693 C0T2AG 67953425 EC50 = 12 nM T37693 CX01CP 67953431 EC50 = 0.19 nM T37693 CX13CH 67953836 EC50 = 0.08 nM T37693 CPTA39 67953837 EC50 = 0.23 nM T37693 C4XKL9 67953838 EC50 = 99 nM T37693 CIHR82 67953851 EC50 = 0.067 nM T37693 CGC79J 67953920 EC50 = 1.2 nM T37693 CI86RD 67956378 Ki = 14.1 nM T37693 C3S6AU 67970610 Ki > 7000 nM T37693 CL4K0D 68160786 Ki = 46 nM T37693 CSIR78 68182311 EC50 = 7.2 nM T37693 C7CSY1 68182368 EC50 = 2.1 nM T37693 CPG5Q9 68278877 Ki > 10000 nM T37693 C30INO 68353389 EC50 = 91 nM T37693 C6BG0N 68555650 EC50 = 1 nM T37693 C8PN7J 68603000 EC50 = 108 nM T37693 C9Q1KW 68603392 EC50 = 82.7 nM T37693 CCQ6V1 68603806 EC50 = 13.6 nM T37693 C8BS2C 68604012 EC50 = 20.1 nM T37693 CN2T0C 68604144 EC50 = 21.3 nM T37693 CJ94SD 68604381 EC50 = 53.1 nM T37693 CGE5X2 68604800 EC50 = 14.1 nM T37693 C45DZE 68604816 EC50 = 71.4 nM T37693 CAN1O3 68741582 Ki = 43960 nM T37693 C46DPY 68742556 Ki = 4110 nM T37693 CZL35B 68904230 Ki = 104.71 nM T37693 CQ27WM 68908007 Ki > 1000 nM T37693 C5GLN7 68908342 Ki = 91.2 nM T37693 C75UTD 68908346 Ki = 1.95 nM T37693 C84XYG 68909935 IC50 = 1 nM T37693 CJVP65 68910242 IC50 = 11.22 nM T37693 C1XPM0 69003787 IC50 = 4.5 nM T37693 CIZD23 69007013 EC50 = 5.4 nM T37693 C0WAL2 69111813 Ki = 27870 nM T37693 CNQH46 69240356 IC50 > 10000 nM T37693 C1CY2U 69307211 EC50 = 17.4 nM T37693 C3XV4P 69472197 Ki = 247 nM T37693 CB9ND1 69474632 Ki = 2113.49 nM T37693 C1L3WU 69474974 Ki = 144 nM T37693 C84XJE 69475608 Ki = 263 nM T37693 C4NM1C 69493574 Ki = 1 nM T37693 CO5VN9 70285091 EC50 = 85 nM T37693 C0YH3T 70677671 Ki > 10000 nM T37693 CQT54O 70677672 Ki > 10000 nM T37693 CR71AY 70677673 Ki = 2450 nM T37693 C8VQ0M 70677674 Ki = 13300 nM T37693 CURQ38 70677675 Ki > 10000 nM T37693 CGR4U7 70677676 Ki > 10000 nM T37693 CFMD45 70677677 EC50 = 92 nM T37693 C2E1AD 70677804 Ki = 5150 nM T37693 CVX9I7 70677805 Ki = 267 nM T37693 CLWV92 70677806 Ki = 1680 nM T37693 CCE2U9 70677807 EC50 = 213 nM T37693 C74KDW 70677808 Ki = 3570 nM T37693 CK4C2I 70677809 Ki = 392 nM T37693 CTYE29 70677810 Ki = 1760 nM T37693 CSGH58 70677953 EC50 = 14 nM T37693 CY3O0R 70677954 Ki = 4800 nM T37693 CCUW05 70677955 Ki = 185 nM T37693 CB4P6Y 70677956 Ki = 1940 nM T37693 C6ESV8 70677957 Ki = 350 nM T37693 C3F2AY 70677958 Ki = 2200 nM T37693 CV7Q3G 70677959 Ki = 4120 nM T37693 C4Y1LE 70678097 Ki = 465 nM T37693 C3DX1U 70678098 Ki = 3010 nM T37693 C71DQG 70678099 EC50 = 54 nM T37693 CJ0P4V 70678100 Ki = 10000 nM T37693 C82PMZ 70678101 Ki = 292 nM T37693 CTB19O 70678102 Ki = 1140 nM T37693 C46QGZ 70678238 EC50 = 48 nM T37693 CBX9D4 70678239 Ki >= 10000 nM T37693 CS7FL4 70678240 Ki = 49 nM T37693 C30LIP 70678241 Ki > 10000 nM T37693 CT1EF6 70678242 Ki > 10000 nM T37693 CO7SP4 70681279 Ki = 4.4 nM T37693 CZ3X4M 70681392 Ki = 33 nM T37693 C0SVD9 70681412 Ki = 73.96 nM T37693 C2MSC9 70683383 Ki = 382 nM T37693 C4YUC3 70684359 Ki = 6540 nM T37693 C3IXK2 70684360 Ki = 16900 nM T37693 CK6NA5 70685024 IC50 = 1.585 nM T37693 C65WEJ 70686524 Ki = 3290 nM T37693 CA4UM9 70687741 IC50 = 167 nM T37693 C8WKV5 70687770 IC50 = 38 nM T37693 CJ0Z2Y 70687771 IC50 = 11 nM T37693 CJ6KE0 70687772 IC50 = 3.5 nM T37693 CJMG21 70689659 Ki = 0.6 nM T37693 C2BA8P 70689660 Ki = 1.1 nM T37693 CSI98P 70689667 Ki = 128 nM T37693 C6UVC8 70689694 IC50 = 1 nM T37693 C3L1HS 70689695 IC50 = 14 nM T37693 CN43EU 70689696 IC50 = 51 nM T37693 CQ95RM 70689788 IC50 = 268 nM T37693 CXO85R 70689820 IC50 = 800 nM T37693 C7UJ0Y 70690691 Ki = 11000 nM T37693 CGOP85 70690692 Ki = 15200 nM T37693 C6K9DE 70690693 Ki = 15400 nM T37693 C8OLN3 70691798 Ki = 1.2 nM T37693 C5XZR6 70691799 Ki = 81 nM T37693 CNGX50 70691826 Ki = 348 nM T37693 CYO5G4 70692838 Ki = 12100 nM T37693 CKDW02 70692839 Ki = 8700 nM T37693 CS63PK 70693593 Ki = 104.71 nM T37693 CL06EQ 70693862 Ki = 2.5 nM T37693 CT7Q5W 70693863 Ki = 6 nM T37693 CW8LU2 70693864 Ki = 3 nM T37693 CY4CH9 70694009 Ki = 119.95 nM T37693 CX2NM7 70694867 Ki = 953 nM T37693 CE7W2O 70694868 Ki = 21200 nM T37693 C1PDK2 70695982 Ki = 377 nM T37693 C6YG8R 70696000 IC50 = 7 nM T37693 C1FU9R 70696001 Ki = 294 nM T37693 C8R3JH 70696105 Ki = 1.2 nM T37693 C2JFU3 70696133 Ki = 922.57 nM T37693 CL6WD5 70696134 Ki > 5000 nM T37693 CUS64H 70864970 EC50 = 33 nM T37693 CN5G3Z 70864972 EC50 = 18 nM T37693 CP6FO8 70865026 EC50 = 995 nM T37693 CA8CQ4 70865076 EC50 = 167 nM T37693 C2PJ1D 70865101 EC50 = 11 nM T37693 C5H8UT 70865109 EC50 > 1000 nM T37693 CUY4E2 70865116 EC50 = 166 nM T37693 CQX01V 70865117 EC50 = 17 nM T37693 CR13JM 70865325 EC50 = 55 nM T37693 C4OK5W 70865326 EC50 = 38 nM T37693 C90OTR 70865329 EC50 = 61 nM T37693 CBTY34 71020062 Ki = 2494.08 nM T37693 CC50UG 71113198 EC50 = 4.3 nM T37693 C1NYW6 71116224 Ki = 1929 nM T37693 CU5NM8 71138232 EC50 = 62 nM T37693 CR12DH 71138284 EC50 = 53.8 nM T37693 CEK26Z 71138285 EC50 = 53.8 nM T37693 CVQ1T2 71308155 EC50 = 29 nM T37693 C83XZQ 71308243 Ki = 11 nM T37693 CY8KL0 71449129 IC50 = 530 nM T37693 CD35HU 71449370 Ki > 1000 nM T37693 CPL4J3 71449371 Ki = 689 nM T37693 C9NHQ5 71449464 Ki = 2.9 nM T37693 CAY6E5 71449465 Ki = 0.3 nM T37693 CF0HK8 71449466 Ki = 1.3 nM T37693 CCYF04 71449467 Ki = 14.8 nM T37693 CDT13U 71449468 Ki = 19.9 nM T37693 CV7SA8 71449529 IC50 > 5000 nM T37693 CHW0A3 71449530 IC50 > 1000 nM T37693 CAYC78 71449541 IC50 > 5000 nM T37693 C0MN4L 71449542 IC50 > 1000 nM T37693 C8P3SF 71449726 Ki = 3.62 nM T37693 CAC5B0 71449939 Ki > 1000 nM T37693 C2S4KP 71449940 Ki > 1000 nM T37693 CM1R0G 71449941 Ki > 1000 nM T37693 C1J9BZ 71449943 Ki > 1000 nM T37693 CWDN02 71450141 Ki = 213 nM T37693 C98YPR 71450142 Ki = 494 nM T37693 CN5SC9 71450187 Ki = 2453 nM T37693 C2S6LQ 71450188 Ki = 1657 nM T37693 C0ZT2Y 71450189 Ki = 20000 nM T37693 CT83NB 71450463 EC50 = 6 nM T37693 C8W2GK 71450464 EC50 = 49 nM T37693 CLDY61 71450465 EC50 = 4.7 nM T37693 C0DG7B 71450466 EC50 = 26 nM T37693 C1EN0J 71450467 EC50 = 106 nM T37693 CYT1Z2 71450516 EC50 = 24 nM T37693 C9S8IF 71450517 EC50 = 41 nM T37693 C2GOT7 71450518 EC50 = 24 nM T37693 CI1L7R 71450519 EC50 = 23 nM T37693 CN96YC 71450520 EC50 = 489 nM T37693 C35AKH 71450521 EC50 > 10000 nM T37693 C1BJ9N 71450522 EC50 = 7892 nM T37693 C9FY0A 71450641 Ki = 152 nM T37693 CZJV01 71450642 Ki = 22 nM T37693 CV90CJ 71450643 Ki = 2.3 nM T37693 CIS2K4 71450921 Ki = 44 nM T37693 C85ANU 71451170 Ki > 3000 nM T37693 C60ILF 71451171 Ki > 1000 nM T37693 C75VXY 71451172 EC50 = 371 nM T37693 CAWS56 71451265 Ki = 7.9 nM T37693 CYU28K 71451266 Ki = 15.2 nM T37693 C90EMT 71451267 Ki = 0.1 nM T37693 CH1QU4 71451268 Ki = 6.5 nM T37693 C7YM3V 71451269 Ki = 13.3 nM T37693 C2D3EN 71451270 Ki = 118.7 nM T37693 CYD6H5 71451324 IC50 > 1000 nM T37693 CI1DG5 71451325 IC50 > 5000 nM T37693 C1EL7T 71451331 IC50 > 5000 nM T37693 C8J1YK 71451332 IC50 > 5000 nM T37693 CDJO69 71451333 IC50 > 5000 nM T37693 C7NS9H 71451521 Ki > 10000 nM T37693 CDES68 71451522 Ki = 1180 nM T37693 CJ7BK4 71451761 Ki > 1000 nM T37693 CB9MI7 71451970 Ki = 5683 nM T37693 CHN2J6 71451971 Ki = 167 nM T37693 CWU40D 71451972 Ki = 35969.96 nM T37693 C6XJ3A 71451973 Ki = 182 nM T37693 C9WSP6 71451974 Ki = 160 nM T37693 C65FUD 71451975 EC50 = 17.08 nM T37693 CE5H8L 71451976 EC50 = 5.73 nM T37693 CVUQ43 71452011 Ki = 1548 nM T37693 C4POZ7 71452013 Ki > 20000 nM T37693 CM8X9C 71452295 EC50 = 46 nM T37693 CROF14 71452296 EC50 = 344 nM T37693 CLW23T 71452368 EC50 = 6.4 nM T37693 CFH25Z 71452369 EC50 = 96 nM T37693 CA8MB6 71452370 EC50 = 3.6 nM T37693 CM17YT 71452371 EC50 = 11 nM T37693 C01EHK 71452372 EC50 = 695 nM T37693 C3WB7F 71452473 Ki = 2.1 nM T37693 CZ65ND 71452474 Ki = 134 nM T37693 CU0C6V 71452475 Ki = 27 nM T37693 CH94DF 71452701 Ki = 2.9 nM T37693 C3M6NR 71452739 IC50 = 410 nM T37693 CA0IP1 71453003 Ki > 3000 nM T37693 CF53WM 71453004 EC50 = 191 nM T37693 C96RTE 71453082 Ki = 5.5 nM T37693 C9SN8B 71453083 Ki = 15.2 nM T37693 CUW47P 71453084 Ki = 0.4 nM T37693 C1S4AY 71453085 Ki > 10000 nM T37693 COV6P0 71453086 Ki = 77.5 nM T37693 CT2AJ3 71453087 Ki = 230 nM T37693 CI13LY 71453088 Ki = 340 nM T37693 C3ND5C 71453142 IC50 > 5000 nM T37693 C5B4UC 71453148 IC50 > 5000 nM T37693 CJ4LV0 71453149 IC50 > 5000 nM T37693 C2R8FM 71453477 Ki = 0.28 nM T37693 C9OS2A 71453478 Ki > 1000 nM T37693 CC25TP 71453584 Ki > 1000 nM T37693 CL1R2P 71453777 Ki = 2636 nM T37693 C58LXU 71453778 Ki = 146 nM T37693 CP86RY 71453779 Ki = 221 nM T37693 CMWD96 71453780 Ki = 595 nM T37693 CYP6M9 71453781 Ki > 20000 nM T37693 CC73DS 71453820 Ki = 5507 nM T37693 C59BKG 71454089 EC50 = 201 nM T37693 CRZ5O1 71454090 EC50 = 47 nM T37693 CEFK54 71454091 EC50 = 394 nM T37693 CC15FR 71454137 EC50 = 101 nM T37693 CI87XN 71454138 EC50 = 74 nM T37693 CC7HZ4 71454139 EC50 = 15 nM T37693 CO2D9I 71454140 EC50 = 1.4 nM T37693 CZE87R 71454141 EC50 = 646 nM T37693 C25MZX 71454142 EC50 = 488 nM T37693 CK1L0A 71454143 EC50 = 939 nM T37693 C7RI0X 71454144 EC50 > 10000 nM T37693 C5TDX4 71454145 EC50 = 14 nM T37693 CXY23Z 71454233 Ki = 1.1 nM T37693 C87ZBR 71454234 Ki = 3.3 nM T37693 CJGD87 71454235 Ki = 38 nM T37693 C6Z9KB 71454236 Ki = 3.2 nM T37693 C4JIA0 71454453 Ki = 505 nM T37693 CCU61Z 71454454 Ki = 5 nM T37693 C1THG2 71454455 Ki = 103 nM T37693 C35CMH 71454823 Ki = 93.9 nM T37693 CK5Z8D 71454824 Ki = 2.5 nM T37693 C1OC6X 71454884 IC50 > 1000 nM T37693 CX36YH 71454885 IC50 > 1000 nM T37693 C2JYF6 71455057 Ki = 1790 nM T37693 C81WIN 71455077 Ki = 3.45 nM T37693 CV5QR7 71455189 Ki > 1000 nM T37693 C6WYJ1 71455190 Ki > 1000 nM T37693 CYI08X 71455304 Ki > 1000 nM T37693 CBM5C8 71455314 Ki > 1000 nM T37693 CDG5V0 71455315 Ki > 1000 nM T37693 CH8S0X 71455316 Ki > 1000 nM T37693 CJ4DG1 71455514 Ki = 688 nM T37693 C0HA7N 71455515 Ki = 3553 nM T37693 CCR74A 71455516 Ki = 158 nM T37693 C7LHZ2 71455517 Ki > 20000 nM T37693 C9OT7E 71455518 Ki = 203 nM T37693 C1LS5H 71455552 Ki = 13947 nM T37693 C2XH7I 71455827 EC50 = 5.4 nM T37693 CFJK21 71455875 EC50 = 4.7 nM T37693 CSHB15 71455876 EC50 = 35 nM T37693 CEJ2T3 71455989 Ki = 192 nM T37693 CM0PT2 71456201 Ki = 13 nM T37693 C5KI1U 71456202 Ki = 60 nM T37693 C68CNX 71456598 Ki = 1.1 nM T37693 CKTP96 71456599 Ki = 957.1 nM T37693 C7HW1G 71456600 Ki = 130 nM T37693 C0QSJ4 71456601 Ki = 19.3 nM T37693 C0NV6W 71456602 Ki > 10000 nM T37693 C9LOZ3 71456650 IC50 > 5000 nM T37693 CNS3L4 71456661 IC50 > 5000 nM T37693 C1D6KG 71456857 Ki > 10000 nM T37693 CP1OY9 71456858 Ki > 10000 nM T37693 CP4K8E 71456859 Ki = 580 nM T37693 COQ29S 71456981 Ki > 1000 nM T37693 C9ZC2I 71457083 Ki > 1000 nM T37693 CI5HK6 71457090 Ki > 1000 nM T37693 C53VGN 71457303 Ki = 18199.98 nM T37693 C42MDX 71457304 Ki > 20000 nM T37693 C1C9FL 71457305 Ki > 20000 nM T37693 CFG6E0 71457306 Ki > 20000 nM T37693 C12OEY 71457307 Ki = 10850 nM T37693 CFNI69 71457308 Ki > 20000 nM T37693 CW79ZE 71457341 Ki = 153 nM T37693 CKWG06 71457342 Ki = 4645 nM T37693 CHF86C 71457343 Ki = 14000 nM T37693 C6AWM3 71457619 EC50 = 56 nM T37693 CID47K 71457677 EC50 = 0.55 nM T37693 C6LYF4 71457678 EC50 = 6.5 nM T37693 COS48L 71457679 EC50 = 3.3 nM T37693 C5G7LZ 71457680 EC50 = 17 nM T37693 CQH74V 71457790 Ki = 31 nM T37693 CS3XD2 71457791 Ki = 1.3 nM T37693 CT90JC 71457792 Ki = 10 nM T37693 CGO45N 71457793 Ki = 536 nM T37693 C0JP3H 71457794 Ki = 2.2 nM T37693 CJ6N5E 71458352 Ki > 3000 nM T37693 CL1KS5 71458353 EC50 = 297 nM T37693 CU4RF3 71458354 Ki > 3000 nM T37693 CM2N8G 71458457 Ki = 139.1 nM T37693 C6S4RO 71458508 IC50 > 5000 nM T37693 CH7L4U 71458714 Ki > 10000 nM T37693 C35XHD 71458715 Ki = 690 nM T37693 C70YWM 71458948 Ki > 1000 nM T37693 C38CRF 71458950 Ki > 1000 nM T37693 C4DFC8 71458951 Ki > 1000 nM T37693 C9SUN1 71459136 Ki = 462 nM T37693 C1L3CZ 71459137 Ki > 20000 nM T37693 C21WTX 71459138 Ki > 20000 nM T37693 CUP6O2 71459139 Ki = 9318.99 nM T37693 C4O9AG 71459140 Ki = 154 nM T37693 CEK2A3 71459141 EC50 = 4.11 nM T37693 CI8N9M 71459142 Ki = 11779.99 nM T37693 CU1YC4 71459143 Ki = 596 nM T37693 CKME06 71459192 Ki = 1713 nM T37693 CGF62Y 71459194 Ki = 948 nM T37693 C51CZF 71459196 Ki > 20000 nM T37693 CT2YD6 71459512 EC50 = 18 nM T37693 CA46PX 71459513 EC50 = 219 nM T37693 CY1HJ8 71459578 EC50 = 129 nM T37693 CSA07B 71459579 EC50 = 38 nM T37693 CI4W2B 71459580 EC50 = 2.5 nM T37693 CNG46Q 71459581 EC50 > 10000 nM T37693 CM8U2X 71459582 EC50 = 95 nM T37693 C4Q3VE 71459583 EC50 = 227 nM T37693 CIS71D 71459709 Ki = 33 nM T37693 CO81NJ 71459905 Ki = 89 nM T37693 C0ZD3W 71459906 Ki = 25 nM T37693 C42XOR 71459907 Ki = 18 nM T37693 CA8SK6 71459922 Ki = 0.032 nM T37693 CUQK68 71459945 IC50 = 1200 nM T37693 C97TBJ 71460194 Ki > 3000 nM T37693 C1K6MS 71460195 Ki = 3639 nM T37693 CU3W9O 71460308 Ki = 7.3 nM T37693 C0GF4X 71460309 Ki = 0.8 nM T37693 CZT47C 71460310 Ki = 16 nM T37693 C4FD5O 71460311 Ki = 0.09 nM T37693 C84SOK 71460312 Ki = 89.1 nM T37693 C4T8BN 71460313 Ki > 10000 nM T37693 CV6C0O 71460352 IC50 = 5000 nM T37693 C1M8KG 71460548 Ki = 265 nM T37693 C8TE6M 71460655 EC50 = 8.3 nM T37693 CNA5B4 71460951 EC50 = 13.42 nM T37693 C6AI9M 71460952 Ki > 20000 nM T37693 CC64PU 71460953 Ki = 22 nM T37693 CVH89E 71460954 Ki = 12550 nM T37693 CWZ13R 71460978 Ki = 5865 nM T37693 C82PAR 71460979 Ki = 8946 nM T37693 C25NCA 71461256 EC50 = 63 nM T37693 CZ94DS 71461257 EC50 = 137 nM T37693 COT0U9 71461320 EC50 = 5.9 nM T37693 CS8Y2Z 71461321 EC50 = 40 nM T37693 C02PKW 71461322 EC50 = 313 nM T37693 CO7MH0 71461323 EC50 = 1421 nM T37693 C40DFP 71461324 EC50 = 103 nM T37693 CP6YI3 71461325 EC50 = 35 nM T37693 CCV94E 71461421 Ki = 278 nM T37693 C09VOG 71461422 Ki = 44 nM T37693 CEM06G 71461910 Ki > 3000 nM T37693 CF9AQ4 71462003 Ki = 31.5 nM T37693 CV9M1I 71462004 Ki = 4.4 nM T37693 C08TZO 71462005 Ki > 10000 nM T37693 CK7FA6 71462047 IC50 > 5000 nM T37693 CVB2R9 71462053 IC50 > 1000 nM T37693 C1VOK3 71462054 IC50 > 5000 nM T37693 CBM3S6 71462240 Ki = 1120 nM T37693 CG16QI 71462668 Ki = 310 nM T37693 CX25GM 71462669 Ki = 101 nM T37693 CR3J4Z 71462670 Ki > 20000 nM T37693 CH67IE 71462671 Ki > 20000 nM T37693 CM27NV 71462714 Ki = 1073 nM T37693 CRNO72 71462715 Ki = 7779 nM T37693 CE7O6K 71462979 EC50 = 209 nM T37693 CG25YZ 71463044 EC50 = 71 nM T37693 C3RK6B 71463045 EC50 = 749 nM T37693 C0U5IW 71463046 EC50 = 897 nM T37693 CU2W0X 71463047 EC50 = 3 nM T37693 CE0BD5 71463048 EC50 = 9.5 nM T37693 CER92U 71463049 EC50 = 35 nM T37693 C6RIO7 71463050 EC50 = 9354 nM T37693 CEO29S 71463152 Ki = 2.8 nM T37693 CG9HX2 71463153 Ki = 174 nM T37693 C1QTI4 71463154 Ki = 10 nM T37693 CH3W2U 71463155 Ki = 19 nM T37693 CP26EI 71539529 Ki = 11 nM T37693 C94GWF 71539530 Ki = 215 nM T37693 C8MFO7 71539582 EC50 = 75 nM T37693 CC7QJ5 71539583 Ki = 22.5 nM T37693 CH16LA 71539584 EC50 = 37 nM T37693 CIY1E4 71539585 EC50 = 53 nM T37693 CDF9S6 71539644 EC50 > 3000 nM T37693 CBS70R 71539645 EC50 = 160 nM T37693 CK7OC8 71539693 Ki = 30 nM T37693 C0KU9T 71539694 EC50 = 27 nM T37693 CCW9X4 71539695 EC50 = 57 nM T37693 C1I8AV 71539696 EC50 = 73 nM T37693 CHM1K5 71539697 EC50 = 49 nM T37693 CKGT70 71539698 EC50 = 46 nM T37693 C7XLD6 71539749 EC50 = 113 nM T37693 C4UN2K 71539750 EC50 = 48 nM T37693 C3E8XT 71539751 EC50 = 42 nM T37693 C6LSP2 71539752 EC50 > 3000 nM T37693 CD8TB3 71539800 EC50 = 106 nM T37693 C6K3BY 71539801 EC50 = 3550 nM T37693 CG3XK5 71539802 EC50 = 76 nM T37693 C5OFT1 71539803 EC50 = 92 nM T37693 CO49HY 71539804 EC50 = 270 nM T37693 CLOM30 71539855 EC50 = 144 nM T37693 CNI32T 71539856 EC50 = 181 nM T37693 CS4O0R 71539907 EC50 = 4300 nM T37693 CD1X8N 71539953 EC50 = 231 nM T37693 C8L6RO 71539954 EC50 = 1760 nM T37693 C9N7YA 71544706 IC50 > 690 nM T37693 C92NEY 71544707 IC50 = 2500 nM T37693 C4N3OC 71545856 IC50 = 500 nM T37693 CV5E9K 71546015 IC50 > 10000 nM T37693 CJ75FS 71546180 IC50 = 5700 nM T37693 C6W5VM 71546181 IC50 > 10000 nM T37693 C5JD2B 71546182 IC50 = 360 nM T37693 CQJE12 71546834 IC50 = 2500 nM T37693 C29NBP 71546835 IC50 = 1200 nM T37693 C1IR3O 71559417 EC50 = 27 nM T37693 C1R6XV 71559418 EC50 = 1.8 nM T37693 CM56QN 71559419 EC50 = 20 nM T37693 C7LK1F 71559522 EC50 = 29 nM T37693 CZYK61 71559523 EC50 = 20 nM T37693 CQ20NX 71559524 EC50 = 16 nM T37693 CP5HX4 71559525 EC50 = 4 nM T37693 C5DRB3 71559526 EC50 = 4.6 nM T37693 CMT2O6 71559637 EC50 = 15 nM T37693 C40KSJ 71559638 EC50 = 55 nM T37693 CEXC24 71559639 EC50 = 22 nM T37693 C10SJV 71559641 EC50 = 7 nM T37693 CK57LU 71561577 Ki = 3.58 nM T37693 C2ZT8O 71562536 Ki = 85 nM T37693 CV6D0B 71562537 Ki = 138 nM T37693 CDOC40 71562538 Ki = 412 nM T37693 C5VMJ8 71562539 EC50 = 587 nM T37693 C9O0IY 71562646 Ki > 10000 nM T37693 CR5DA3 71562647 Ki > 10000 nM T37693 C8Q3TG 71562648 Ki = 325 nM T37693 CJH90S 71562649 Ki = 956 nM T37693 CW8UR7 71562650 Ki > 10000 nM T37693 CDL5T4 71562651 Ki > 10000 nM T37693 CVW4E9 71562652 Ki = 372 nM T37693 CFU7J4 71562780 Ki = 10.6 nM T37693 CFC4X3 71562781 Ki = 11.2 nM T37693 C8XO4U 71562782 Ki = 9.51 nM T37693 CBQ4R3 71562784 Ki = 212 nM T37693 C8WGI2 71562897 Ki = 524 nM T37693 CCZ60L 71562898 Ki > 10000 nM T37693 CD37US 71562899 Ki > 10000 nM T37693 CV8Y9G 71562900 Ki = 3652 nM T37693 CUIY12 71562901 Ki = 469 nM T37693 CIX50M 71562902 Ki = 37 nM T37693 CF0HO4 71563025 Ki = 3526 nM T37693 C6PKB2 71563026 Ki = 363 nM T37693 CNG41L 71563027 Ki = 237 nM T37693 CR9X5F 71563028 Ki = 103 nM T37693 CJE6L8 71563029 Ki = 11.6 nM T37693 CBN0L8 71563030 Ki > 10000 nM T37693 C6T1CA 71563145 Ki > 10000 nM T37693 CMGT96 71563146 Ki = 3620 nM T37693 CE7M3O 71563147 Ki = 2830 nM T37693 C6TK3A 71563148 Ki = 8.74 nM T37693 CM48BC 71563149 Ki = 18.5 nM T37693 CY6IM3 71563150 Ki = 21 nM T37693 CG4K6V 71563277 Ki = 12.3 nM T37693 CC31QD 71563278 Ki = 6.95 nM T37693 CZ7FL2 71563279 Ki = 1.12 nM T37693 C9M8XO 71563280 Ki = 3.27 nM T37693 C98DXW 71563282 Ki = 20 nM T37693 CJK19B 71580293 IC50 = 0.58 nM T37693 CPB6D8 71580820 Ki = 333 nM T37693 C1WH2Q 71580821 Ki = 114 nM T37693 C80PME 71580822 Ki = 588 nM T37693 CSH40Y 71580902 Ki = 2.5 nM T37693 CIU39D 71583195 Ki = 490 nM T37693 CS21CO 71583291 Ki = 2943 nM T37693 C89NPS 71583306 Ki = 3855 nM T37693 C3PEF1 71583307 Ki = 276 nM T37693 CG6VC9 71583308 Ki = 214 nM T37693 CZW69O 71583309 Ki = 609 nM T37693 C6ST9V 71583310 Ki = 1310 nM T37693 C6FDX7 71583311 Ki = 89 nM T37693 CX0JF3 71583401 Ki = 458.2 nM T37693 CS52BT 71583402 Ki > 40000 nM T37693 CNAX48 71583403 Ki > 40000 nM T37693 C3LND0 71583404 Ki > 10000 nM T37693 CM09HD 71583405 Ki > 40000 nM T37693 C9IY5E 71583419 Ki = 88 nM T37693 C2D4XJ 71583420 Ki = 16 nM T37693 CS9CT6 71583421 IC50 = 13 nM T37693 C8GT1B 71583422 Ki = 42 nM T37693 CKG49Z 71583423 Ki = 72 nM T37693 C79HPR 71583424 Ki = 12 nM T37693 C5Q1DF 71583425 Ki = 768 nM T37693 C7BTX6 71583521 Ki > 10000 nM T37693 C78ZRD 71583522 Ki = 18220 nM T37693 C94AJQ 71583523 Ki > 40000 nM T37693 C30RXC 71583524 Ki > 10000 nM T37693 C9C2YD 71583608 Ki = 83.95 nM T37693 CPC06E 71583609 Ki = 25 nM T37693 CQBV09 71583610 Ki = 172.98 nM T37693 C35QNI 71583711 Ki = 137 nM T37693 C7DET3 71583712 Ki = 46.99 nM T37693 CLTK19 71583713 Ki = 19 nM T37693 CK5DX1 71583714 Ki = 457 nM T37693 C30KRJ 71583715 Ki = 34.99 nM T37693 CTN97S 71583827 Ki = 638 nM T37693 C1K7LR 71583828 Ki = 38 nM T37693 CM9N3D 71583829 Ki = 59.98 nM T37693 CU1QP7 71583830 Ki = 2745 nM T37693 CBN2W1 71583831 Ki = 2301.44 nM T37693 CX5MC7 71583832 Ki = 13000 nM T37693 CCKZ69 71583941 Ki = 5188 nM T37693 C83XPV 71583942 Ki > 20000 nM T37693 CCPT98 71583943 Ki = 1101 nM T37693 C2NB8E 71583944 Ki = 6740 nM T37693 CC91ZV 71583945 Ki = 272.9 nM T37693 CSF72V 71583946 Ki = 680 nM T37693 C8EZF9 71584045 Ki = 1312 nM T37693 CQ86ER 71584046 Ki = 696 nM T37693 C86ZXK 71584047 Ki = 1279.38 nM T37693 CTYS72 71584048 Ki = 211.84 nM T37693 CEGV60 71584049 Ki > 20000 nM T37693 CNWE02 71584050 Ki = 12.62 nM T37693 CKB0G2 71584155 Ki = 72.95 nM T37693 CED16K 71584156 Ki = 35.97 nM T37693 CD9QX6 71584157 Ki = 14 nM T37693 CJQY30 71584158 Ki = 36.98 nM T37693 CJ58HL 71584159 Ki = 2.799 nM T37693 CYHF59 71584160 Ki = 221.82 nM T37693 C4TL1Z 71584275 Ki = 136 nM T37693 CLZX28 71584276 Ki = 164 nM T37693 CE7A4L 71584277 Ki = 3.396 nM T37693 C3ILW7 71584278 Ki = 5.598 nM T37693 CF4RV8 71584279 Ki = 2.999 nM T37693 C2W1IH 71584410 Ki = 5.395 nM T37693 CZH52F 71584411 Ki = 5.794 nM T37693 CI0E4G 71584412 Ki = 4.295 nM T37693 C6C8TB 71584413 Ki = 71.94 nM T37693 CV26EB 71584414 Ki = 106.91 nM T37693 C0T9US 71584415 Ki = 221.82 nM T37693 CMYO23 71587360 EC50 = 10.9 nM T37693 C5YQ2V 71599710 EC50 = 0.78 nM T37693 C7KSG0 71621165 Ki = 10.9 nM T37693 C0Z5QS 71623175 Ki = 44 nM T37693 CYF3V8 71623176 Ki = 174 nM T37693 CWN27F 71623177 Ki = 230 nM T37693 C9PND6 71623178 Ki = 130 nM T37693 CW1R4X 71623179 Ki = 130 nM T37693 C9XKY7 71623225 Ki = 280 nM T37693 C4PQY5 71623226 Ki = 470 nM T37693 C5AX6I 71623227 Ki = 71 nM T37693 C7W6YB 71623228 Ki = 46 nM T37693 CZ0N7J 71623229 Ki = 94 nM T37693 C6NR2Q 71623230 Ki = 577 nM T37693 CY3SR4 71623284 Ki = 190 nM T37693 C8Z4IE 71623285 Ki = 166 nM T37693 CREW95 71623286 Ki = 3600 nM T37693 CGQD80 71623287 Ki = 120 nM T37693 CJF0C2 71623288 Ki = 540 nM T37693 CV1YU9 71623289 Ki = 210 nM T37693 CGI80R 71623340 Ki = 230 nM T37693 C1I8WY 71623341 Ki = 150 nM T37693 C7BHC6 71623342 Ki = 262 nM T37693 CG9X8V 71623343 Ki = 73 nM T37693 C03LQH 71623344 Ki = 102 nM T37693 CO2CQ4 71623345 Ki = 170 nM T37693 CN7VC0 71624052 Ki = 53 nM T37693 CJ67PB 71624053 Ki = 680 nM T37693 C3FNI8 71624054 Ki = 166 nM T37693 CO8RP5 71624055 Ki = 390 nM T37693 CBS46L 71624056 Ki = 120 nM T37693 C1G8AO 71624057 Ki = 34 nM T37693 CS3J0O 71624058 Ki = 9.5 nM T37693 CAMI85 71624059 Ki = 14 nM T37693 CRY61V 71624060 Ki = 5.5 nM T37693 CXS93U 71624177 Ki = 14 nM T37693 C46VIA 71624178 Ki = 36 nM T37693 CAQ3Z2 71624179 Ki = 66 nM T37693 CZR79M 71624180 EC50 = 2.5 nM T37693 C83JIM 71624181 Ki = 30 nM T37693 CUD56P 71624182 Ki = 20 nM T37693 C80NJP 71624301 Ki = 18 nM T37693 C85TFY 71624302 Ki = 31 nM T37693 CU1I6J 71624303 Ki = 75 nM T37693 CO3LE7 71624304 Ki = 55 nM T37693 C3O7BW 71624305 Ki = 4 nM T37693 C28SIU 71624306 Ki = 310 nM T37693 CS72QZ 71624432 Ki = 140 nM T37693 CJ57PR 71624543 Ki = 32 nM T37693 C45ZCL 71656839 Ki = 26.5 nM T37693 C3P7BM 71656931 Ki = 281 nM T37693 C6LF7K 71660058 Ki > 5000 nM T37693 CAY05V 71660059 Ki = 66 nM T37693 CSI3T7 71660060 Ki = 16 nM T37693 C3ESZ4 71660061 Ki = 17 nM T37693 CHNS93 71660062 Ki = 204 nM T37693 CW06JB 71660102 Ki > 5000 nM T37693 CVGZ69 71660103 Ki = 0.9 nM T37693 CXFA37 71660104 Ki = 8 nM T37693 C13HSU 71660105 Ki = 209 nM T37693 CJ01PU 71660182 Ki = 147 nM T37693 C6QNX4 71661529 Ki = 338 nM T37693 CS4OT0 71661531 Ki = 5.5 nM T37693 CA64ZQ 71661713 Ki = 9 nM T37693 CE24RP 71661714 Ki = 40.5 nM T37693 CW1U6C 71661715 Ki = 671.8 nM T37693 CB9FL3 71661716 Ki = 11.3 nM T37693 CXER89 71661717 Ki = 261.7 nM T37693 CGI7V1 71661718 Ki = 100.3 nM T37693 CR9NG5 71661887 Ki = 67.2 nM T37693 CET75O 71661888 Ki = 11.2 nM T37693 C60UIK 71661889 Ki = 33.3 nM T37693 CO34HE 71661890 Ki = 121.2 nM T37693 CY8V6D 71661891 Ki = 7.8 nM T37693 CM86BY 71662072 Ki = 365.3 nM T37693 C8GR6J 71662073 Ki = 49.2 nM T37693 CH0E7F 71662074 Ki = 14 nM T37693 C65QMB 71662076 Ki = 46.7 nM T37693 CG36WL 71662252 Ki = 63.5 nM T37693 C5S1CO 71662414 Ki = 338 nM T37693 C3E1AR 71662416 Ki = 551 nM T37693 C7N2BM 71680717 Ki = 0.84 nM T37693 CJK5C9 71680718 Ki = 12.3 nM T37693 CB7N4D 71680719 Ki = 7.22 nM T37693 CZ2OI1 71680720 Ki = 4.95 nM T37693 CTHM04 71680721 Ki = 42 nM T37693 CE1IJ5 71680722 Ki = 31 nM T37693 C14BYK 71680878 Ki = 2.56 nM T37693 CY1ZL3 71680879 Ki = 40 nM T37693 C2EMP9 71680880 Ki = 8.93 nM T37693 C9ECU3 71680881 Ki = 2.86 nM T37693 C3HR1X 71680882 Ki = 57 nM T37693 C5AYI9 71681038 Ki = 10.3 nM T37693 CQI90H 71681039 Ki = 3.41 nM T37693 CFBR90 71681040 Ki = 47 nM T37693 CVW58F 71681041 Ki = 10.3 nM T37693 C0SOY4 71681042 Ki = 6.21 nM T37693 C12PXS 71681193 Ki = 55 nM T37693 C3KQZ0 71681194 Ki = 6.31 nM T37693 C0S3LB 71681195 Ki = 3.88 nM T37693 CY6AJ7 71681196 Ki = 52 nM T37693 C5K9FS 71681197 Ki = 37 nM T37693 CXC1Y5 71681346 Ki = 30 nM T37693 CCO9K8 71681347 Ki = 98 nM T37693 C6WQ9U 71681348 Ki = 9.52 nM T37693 C3HUW6 71681349 Ki = 6.57 nM T37693 C9LV4D 71681350 Ki = 4.92 nM T37693 CVB7N1 71681500 Ki = 10.1 nM T37693 C5D8CU 71681501 Ki = 6.24 nM T37693 C0JVS9 71681502 Ki = 15 nM T37693 CMWR71 71681503 Ki = 11.6 nM T37693 CWQ86H 71681504 Ki = 220 nM T37693 C6MKX3 71681665 Ki = 181 nM T37693 CB63MS 71681666 Ki = 350 nM T37693 CDJH76 71682490 Ki = 6830 nM T37693 C48BSN 71682637 Ki = 795 nM T37693 C0O9HE 71682639 Ki = 338 nM T37693 CZE6R2 71682640 Ki = 1770 nM T37693 C2FBL9 71682641 Ki = 3420 nM T37693 CTOL05 71682642 Ki = 1480 nM T37693 CDX59H 71682795 Ki = 444 nM T37693 C3S1OE 71682796 Ki = 660 nM T37693 CNM1Y8 71682797 Ki = 1560 nM T37693 C0HS4I 71682799 Ki = 578 nM T37693 C12BCL 71682928 Ki = 22 nM T37693 CK0Y3J 71682950 Ki = 578 nM T37693 C1AI4R 71683077 Ki = 10.3 nM T37693 CHZ86D 71683078 Ki = 12.7 nM T37693 C2WK8I 71683079 Ki = 358 nM T37693 C9RZG6 71683080 Ki = 106 nM T37693 CGFD28 71683081 Ki = 10.4 nM T37693 C7WYZ1 71683082 Ki = 5.22 nM T37693 CMBN92 71683085 Ki = 0.81 nM T37693 CUZ0W2 71717393 Ki = 9.83 nM T37693 CM9RY4 71719542 EC50 = 490 nM T37693 CD4P1K 71720085 Ki = 750 nM T37693 C1E9DF 71720136 EC50 = 22 nM T37693 C1FYA8 71720426 IC50 = 300 nM T37693 CM4Y5J 71720818 Ki = 42 nM T37693 C87UKF 71761847 EC50 = 97.4 nM T37693 COW3E7 71762083 EC50 = 82.4 nM T37693 C5BMG6 71764824 EC50 = 4.5 nM T37693 C37SCL 71769055 Ki > 1000 nM T37693 C3N8JE 71769056 Ki > 1000 nM T37693 CRFW13 71769176 EC50 = 2.56 nM T37693 CP7HJ4 71769177 Ki > 1000 nM T37693 CEND89 71769178 EC50 = 2.2 nM T37693 CLH7R3 71769179 EC50 = 2.88 nM T37693 C9MGJ3 71769180 EC50 = 2.9 nM T37693 CM14GO 71769181 EC50 = 3.4 nM T37693 CP18RI 71769302 Ki > 1000 nM T37693 CDY27C 71769303 Ki > 1000 nM T37693 C7XW5O 71769304 Ki > 1000 nM T37693 CUOD35 71769305 Ki > 1000 nM T37693 CV2ZY6 71769306 EC50 = 14.8 nM T37693 C4I9VG 71769415 Ki > 1000 nM T37693 C7KC5H 71769416 EC50 = 4.4 nM T37693 C58UGJ 71769417 EC50 = 2.1 nM T37693 C0UEZ7 71769418 EC50 = 1.9 nM T37693 CXHB14 71769420 EC50 = 11.1 nM T37693 C6S8AW 71769535 EC50 = 1.8 nM T37693 CP7V2H 71769536 Ki > 1000 nM T37693 CZC56H 71769537 Ki > 3000 nM T37693 CNHU23 71769538 Ki > 3000 nM T37693 CLDV17 71769539 Ki > 1000 nM T37693 C28WOC 71769540 Ki = 22.1 nM T37693 C8PI3J 72696659 Ki = 367 nM T37693 C1C6NV 72696785 Ki = 1100 nM T37693 CGH72I 72696786 Ki = 990 nM T37693 C05CDA 72696789 Ki = 486 nM T37693 CJEP26 72696921 Ki = 33 nM T37693 C5F1PV 72696922 Ki = 195 nM T37693 CX9S4J 72696925 Ki = 96 nM T37693 C5WLZ7 72697067 Ki = 584 nM T37693 CV0A9W 72697216 Ki = 5.8 nM T37693 C3GZO0 72697217 Ki = 41 nM T37693 COTL98 72697360 Ki = 291 nM T37693 CH9B4Q 72697361 Ki = 377 nM T37693 CAD43M 72697362 Ki = 476 nM T37693 CM6E8A 72697363 Ki = 858 nM T37693 CD3GB6 72697364 Ki = 1800 nM T37693 C0EI4K 72697506 Ki = 559 nM T37693 C0ELS4 72713000 Ki = 10649 nM T37693 CIA04R 72713195 Ki = 835 nM T37693 C4GL6T 72713198 Ki = 89.5 nM T37693 C41DNA 72713406 Ki = 215 nM T37693 C1Z8XN 72713407 Ki = 569 nM T37693 CLO9N1 72713633 Ki = 4501 nM T37693 C5Z7JD 72714381 IC50 = 90 nM T37693 COS7P3 72714471 IC50 > 10000 nM T37693 C5UDE2 72714472 IC50 = 2190 nM T37693 C1ULX5 72714474 EC50 > 10000 nM T37693 CPCW35 72714476 IC50 = 746 nM T37693 C6O0TP 72714569 EC50 > 10000 nM T37693 CZHT65 72714571 IC50 > 10000 nM T37693 C1UVK7 72715369 EC50 = 793 nM T37693 CG76DM 72715370 IC50 > 10000 nM T37693 CTY74C 72715372 EC50 = 103 nM T37693 CWZ3M4 72715374 EC50 > 10000 nM T37693 C86BMU 72715375 EC50 > 10000 nM T37693 C1OHD4 72715447 IC50 = 61 nM T37693 CJHR59 72715448 IC50 = 807 nM T37693 CYPK25 72715612 EC50 > 10000 nM T37693 C5PL4U 72715613 EC50 > 10000 nM T37693 CZ5G1H 72715614 EC50 > 10000 nM T37693 CSBN82 72715615 EC50 = 144 nM T37693 C4XTS1 72715697 EC50 = 245 nM T37693 C7B2VP 72941840 Ki = 1.585 nM T37693 CUA89W 72946872 IC50 = 1.4 nM T37693 C9VFH8 72948608 Ki = 35.6 nM T37693 C91XBO 72948609 Ki = 65 nM T37693 C0MJ4P 72948610 Ki = 16.4 nM T37693 CI43RQ 72948611 Ki = 2.7 nM T37693 CWC76H 72950702 Ki = 0.79 nM T37693 CFID82 72950851 Ki = 3665 nM T37693 C27BSA 72950872 Ki = 1 nM T37693 C7U5EY 72950873 Ki = 4.22 nM T37693 CW83DK 73213196 Ki > 10000 nM T37693 C6K3XI 73293894 EC50 = 5.32 nM T37693 C3F1SC 73293895 Ki = 15.3 nM T37693 C3YO8Q 73293896 EC50 = 11.56 nM T37693 CHK2T9 73293897 EC50 = 17.19 nM T37693 C3R5YW 73293898 EC50 = 10.09 nM T37693 CX1H7E 73346065 EC50 = 4.8 nM T37693 CAW5C0 73346555 Ki = 2169 nM T37693 C1S8UL 73348032 Ki = 2833 nM T37693 CM6OW8 73348033 Ki = 1093 nM T37693 CHZ7J6 73348039 Ki = 519 nM T37693 CDR90N 73348040 Ki = 249 nM T37693 CA1LE3 73349576 Ki = 1313 nM T37693 CQH3O9 73349577 Ki = 73 nM T37693 C8VOI2 73349578 EC50 = 7.3 nM T37693 C5RH9V 73351135 Ki = 502 nM T37693 C2MO1G 73351137 Ki = 370 nM T37693 C6U1IC 73351138 Ki = 740 nM T37693 C28PLQ 73352191 Ki = 600 nM T37693 CL7N1O 73352608 Ki = 827 nM T37693 CQX65M 73352609 Ki = 2690 nM T37693 C9JT1Q 73353637 Ki > 50000 nM T37693 C8R4HE 73354101 Ki = 398 nM T37693 C2N1ZX 73354104 Ki = 521 nM T37693 CG9F2T 73354105 Ki = 264 nM T37693 CALG02 73354922 Ki = 4.56 nM T37693 CYMZ04 73355622 Ki = 1392 nM T37693 CM1R2U 73357166 Ki = 1927 nM T37693 C2I5OW 73357171 Ki = 96 nM T37693 CMO8I2 73357172 Ki = 88 nM T37693 CSND94 73357173 Ki = 3376 nM T37693 CC9J1O 73387573 Ki = 7.7 nM T37693 CV32SE 76309966 EC50 = 22.8 nM T37693 CC0Q2K 76310144 Ki = 3.7 nM T37693 CN4CY1 76310146 Ki = 3 nM T37693 C7T4EN 76310302 Ki > 10000 nM T37693 C0XBS8 76310303 Ki = 863 nM T37693 CRDT21 76310304 Ki > 10000 nM T37693 CUKW03 76310494 Ki = 1832 nM T37693 CWP1I7 76310495 Ki = 4.8 nM T37693 C70IVL 76310496 Ki = 5.1 nM T37693 CZCX06 76310497 Ki = 1 nM T37693 C2REF3 76310520 Ki = 13.7 nM T37693 C1JRI4 76310521 Ki = 594 nM T37693 CG3D6K 76310535 EC50 = 991 nM T37693 CV13PU 76310709 Ki = 240 nM T37693 C1ORB8 76310724 IC50 = 6080 nM T37693 CQR92A 76313974 Ki > 10000 nM T37693 CH8K9Z 76313975 Ki > 10000 nM T37693 CHKE18 76313976 Ki > 5000 nM T37693 CKJ58T 76314156 Ki = 583 nM T37693 C4C3HN 76314157 Ki = 65 nM T37693 CT9X1Q 76314180 Ki = 4.2 nM T37693 C0X5AU 76314195 EC50 > 17000 nM T37693 CI38KM 76314347 IC50 = 5030 nM T37693 CSL9B8 76317193 EC50 = 4.6 nM T37693 C4C2UQ 76317374 Ki = 51.5 nM T37693 CRF5Y3 76317376 Ki = 6.3 nM T37693 CIJ3R1 76317524 Ki = 1526 nM T37693 CNH7R5 76317725 Ki = 2.2 nM T37693 C7NL6Z 76317738 Ki = 7.9 nM T37693 C8R9KD 76317739 Ki = 187 nM T37693 CVI1O0 76317755 EC50 = 9.9 nM T37693 CRF6T0 76317756 EC50 = 84 nM T37693 C1YVQ3 76317757 EC50 = 24.6 nM T37693 CGI2O5 76317912 Ki = 3510 nM T37693 C1I2UO 76317913 Ki = 2000 nM T37693 CE5M1O 76317914 Ki > 10000 nM T37693 CQC2I9 76317932 IC50 = 20000 nM T37693 CO4IL2 76317959 Ki = 10600 nM T37693 CPF5Y0 76320912 Ki = 4.5 nM T37693 CRPD48 76321243 Ki > 5000 nM T37693 C1L5EW 76321244 Ki > 3000 nM T37693 C8S1FB 76321458 EC50 = 165 nM T37693 C04ELZ 76321459 EC50 = 256 nM T37693 CO5LP6 76321460 EC50 = 45 nM T37693 CI2F6O 76321461 EC50 = 1.9 nM T37693 C20OWQ 76321462 EC50 = 236 nM T37693 C4M8ZY 76321622 Ki = 1300 nM T37693 CSXH87 76321623 Ki = 240 nM T37693 CLS36H 76321951 Ki = 3.3 nM T37693 CZ0AS4 76324747 Ki = 1.7 nM T37693 CMP3Z8 76324864 Ki > 10000 nM T37693 CX2F4H 76325028 Ki > 10000 nM T37693 CBLG65 76325060 EC50 = 256 nM T37693 CE3YU9 76325061 EC50 = 1255 nM T37693 C3NB1K 76325062 EC50 = 1973 nM T37693 C0HA3K 76325063 EC50 > 17000 nM T37693 C1W8HB 76325234 Ki = 400 nM T37693 CO05NW 76325235 Ki = 5000 nM T37693 CR2LF5 76325256 IC50 = 1510 nM T37693 C5GI9Z 76325292 Ki > 10000 nM T37693 CN4D3M 76328423 Ki = 801 nM T37693 CSQ0H6 76328424 Ki > 10000 nM T37693 CFGB61 76328601 Ki = 397 nM T37693 CWIF86 76328602 Ki > 10000 nM T37693 CI0SB5 76328619 Ki = 396 nM T37693 C91YWU 76328633 EC50 = 443 nM T37693 C3BZ6H 76328634 EC50 = 1104 nM T37693 C1LN2I 76328635 EC50 = 6.3 nM T37693 CX31IO 76328636 EC50 = 43 nM T37693 C5AV9G 76328789 Ki = 5400 nM T37693 C4QH5I 76328790 Ki = 90 nM T37693 C30AMV 76328791 Ki = 9000 nM T37693 CB1KJ6 76328792 Ki = 500 nM T37693 CJIF43 76328811 IC50 = 1930 nM T37693 CR6IJ1 76331611 Ki = 672 nM T37693 CPV9G7 76331637 IC50 = 168 nM T37693 CBE63L 76331817 Ki = 2.8 nM T37693 CK20OT 76332105 Ki > 10000 nM T37693 CDUQ61 76332106 Ki = 2637 nM T37693 CHV15W 76332282 Ki = 104 nM T37693 CU4B7F 76332298 Ki = 2.8 nM T37693 CT5GH7 76332299 Ki = 481 nM T37693 C9H2JW 76332300 Ki = 80 nM T37693 CTDG64 76332315 EC50 = 40 nM T37693 C6CI5P 76332316 EC50 = 14.7 nM T37693 CJD08P 76335394 EC50 = 4.1 nM T37693 CHRV01 76335726 Ki > 10000 nM T37693 C73ZEL 76335925 Ki > 10000 nM T37693 CSF2G0 76335926 Ki = 1.2 nM T37693 C8ZW2C 76335938 Ki = 63 nM T37693 CFP9L2 76335946 EC50 = 1437 nM T37693 CTG51J 76336093 Ki > 10000 nM T37693 CBVR96 76336107 IC50 = 4090 nM T37693 C6DA9V 77529583 Ki > 10000 nM T37693 C48YMX 84382039 Ki = 23.09 nM T37693 CGTW96 84820114 EC50 = 630 nM T37693 CQE10H 85468767 Ki > 10000 nM T37693 CA0Y8G 85469571 Ki = 4030 nM T37693 C79HPW 86288867 Ki = 52 nM T37693 C98LWE 86669644 EC50 = 32.9 nM T37693 CW3TR2 86669645 EC50 = 2.1 nM T37693 C6ZWO8 86669647 EC50 = 18.5 nM T37693 CU98CB 86669673 EC50 = 0.7 nM T37693 CBP12Z 86688562 EC50 = 0.9 nM T37693 C5PLO7 86688563 EC50 = 24.8 nM T37693 CISP51 86688570 EC50 = 75.6 nM T37693 C1R3AM 87312657 Ki = 6237 nM T37693 CIW56T 88530818 EC50 = 4.7 nM T37693 CV82BP 88530819 EC50 = 130 nM T37693 CY5MX1 89044257 EC50 = 27 nM T37693 C6WZH9 89044294 EC50 = 34 nM T37693 CCU4M3 89994946 Ki = 0.2 nM T37693 CSY12U 89994947 Ki = 1.8 nM T37693 CY9P6G 89994948 Ki = 4.5 nM T37693 CK2DP6 89994949 Ki = 0.7 nM T37693 CHE7R4 89994956 Ki > 10000 nM T37693 C1AP6L 89994960 Ki = 0.7 nM T37693 CLNO80 89994961 Ki = 2.8 nM T37693 CKRG03 89994964 Ki = 1 nM T37693 CJWM12 89994976 Ki = 0.7 nM T37693 C2D8VG 89994977 Ki = 34.5 nM T37693 C3E6HV 89994978 Ki = 1.5 nM T37693 C3BA4K 89994979 Ki = 2.9 nM T37693 CPR34G 89994980 Ki = 0.8 nM T37693 C27XBQ 89994981 Ki = 0.6 nM T37693 C1X9RL 89994983 Ki = 1.4 nM T37693 CU4T7I 89994985 Ki = 1.3 nM T37693 C0CT2S 89994988 Ki = 0.9 nM T37693 C7K6WN 89995197 Ki > 1000 nM T37693 C5QCL7 89995201 Ki = 94 nM T37693 CHZ6G1 90001613 Ki > 1000 nM T37693 C2HLG9 90654966 Ki = 23.1 nM T37693 CE1YD6 90654967 Ki = 0.032 nM T37693 CBG40L 90654968 EC50 = 0.26 nM T37693 CNT15S 90654969 EC50 = 0.7 nM T37693 CV05HR 90654970 EC50 = 21 nM T37693 C7C2EW 90654971 EC50 = 2 nM T37693 CHN43D 90654972 EC50 = 32 nM T37693 CVY83X 90667465 Ki = 2580 nM T37693 C85BUR 90667466 Ki > 10000 nM T37693 C0FZU2 90667467 Ki > 10000 nM T37693 C4MF8A 90667653 Ki > 10000 nM T37693 CR2WI4 90667654 Ki = 1110 nM T37693 C8N0LA 90667655 Ki > 10000 nM T37693 CU23VX 90667656 Ki = 950 nM T37693 CR8I5E 90667657 Ki > 10000 nM T37693 CI61LD 90667658 Ki >= 10000 nM T37693 C7P2EG 90667659 Ki > 10000 nM T37693 CS5DZ4 90667660 Ki = 1810 nM T37693 C31ZMH 90667661 Ki > 10000 nM T37693 CT37YL 90667662 Ki = 980 nM T37693 CJ7V0Y 90667663 Ki = 1560 nM T37693 C54BTS 90667664 Ki > 10000 nM T37693 CJP21Z 90667665 Ki > 10000 nM T37693 C9RM7U 90667666 Ki > 10000 nM T37693 CWS6G3 91824816 Ki = 529 nM T37693 CL7S4U 91844670 EC50 > 10000 nM T37693 C1MB3D 92279023 Ki > 10000 nM T37693 C5J8EZ 101609852 Ki > 10000 nM T37693 CQS1P5 101882735 Ki = 0.12 nM T37693 CHSE20 101882736 Ki = 1.26 nM T37693 C7IP2A 101882737 Ki = 1.47 nM T37693 C0G8PM 101884092 EC50 = 3311 nM T37693 C1FMO9 101884564 Ki = 560 nM T37693 C9ED8P 101884565 Ki = 1270 nM T37693 CHQ86Y 101884566 Ki = 810 nM T37693 CAM2R6 101884567 IC50 > 10000 nM T37693 C5P8CV 101884568 Ki > 10000 nM T37693 CX08DR 101884569 Ki = 1320 nM T37693 C0CB8R 101884572 Ki = 2560 nM T37693 CNA2H8 101884573 Ki > 10000 nM T37693 CLYG63 101884574 Ki > 10000 nM T37693 CF1D6S 101898797 Ki = 7.36 nM T37693 C2POM8 101898798 Ki = 127.8 nM T37693 C58ZBN 102506267 Ki = 30 nM T37693 CEM4P9 102506268 Ki = 3274 nM T37693 CQF3M5 102514739 Ki = 0.39 nM T37693 CW5RS9 108477332 EC50 = 590 nM T37693 COF7T3 109112982 EC50 > 10000 nM T37693 CYT61B 117698842 EC50 = 26 nM T37693 CSOG62 117776889 EC50 > 3000 nM T37693 C41NLJ 117911680 Ki = 49800 nM T37693 C1Z9RI 118323944 EC50 > 10000 nM T37693 CS6A0V 118323946 EC50 = 4100 nM T37693 CO1I2G 118323957 EC50 > 10000 nM T37693 CP19AD 118323960 EC50 = 458 nM T37693 C4ANZ8 118323971 EC50 = 2380 nM T37693 C1TDN2 118323981 EC50 > 10000 nM T37693 CKN63V 118323997 EC50 = 200 nM T37693 COH45S 118323999 EC50 > 10000 nM T37693 CN4E6J 118324004 EC50 = 8630 nM T37693 C5JAE7 118324005 EC50 > 10000 nM T37693 CU6IQ3 118324016 EC50 = 240 nM T37693 CQC1A2 118324032 EC50 = 6500 nM T37693 CB0IA3 118324050 EC50 = 8690 nM T37693 CF1MC2 118324059 EC50 > 10000 nM T37693 C3KYS6 118324079 EC50 > 10000 nM T37693 CC2KB9 118324098 EC50 > 10000 nM T37693 CMHK20 118324101 EC50 > 10000 nM T37693 CQ7A3N 118324116 EC50 > 10000 nM T37693 CT6GJ1 118324120 EC50 = 61 nM T37693 C6EZ9B 118324131 EC50 > 10000 nM T37693 CQH25F 118324141 EC50 > 10000 nM T37693 CTX50R 118329986 EC50 = 3650 nM T37693 CQD27U 118329991 EC50 > 10000 nM T37693 CLQ6D2 118329993 EC50 = 6700 nM T37693 CE30FQ 118329995 EC50 = 61 nM T37693 CX73EZ 118418641 Ki = 465.9 nM T37693 CNE79D 118418642 EC50 = 1291.4 nM T37693 C79KUR 118418663 EC50 = 47 nM T37693 CBP7X6 118418664 EC50 = 66.8 nM T37693 C5MF1Z 118418666 EC50 = 4.4 nM T37693 CR6D5X 118418701 Ki = 2.5 nM T37693 CUB40K 118418707 EC50 = 444.3 nM T37693 C65EZC 118418720 EC50 = 280.9 nM T37693 CZS8O4 118420675 EC50 = 174.6 nM T37693 C4NQ0D 118420969 EC50 = 2889.7 nM T37693 CR3JE2 118421125 EC50 = 175.6 nM T37693 C8LK9I 118421129 Ki = 416.1 nM T37693 CZ7C5S 118577928 Ki = 26.1 nM T37693 C2TF0N 118577933 Ki = 10.4 nM T37693 C0B3LV 118577936 Ki = 7.7 nM T37693 CIJF40 118577937 Ki = 0.62 nM T37693 CJ1HD0 118577940 Ki = 18.8 nM T37693 CQK7V8 118577942 Ki = 1365 nM T37693 CW3C2E 118577959 Ki = 4.3 nM T37693 CFUY17 118577977 Ki > 3000 nM T37693 CGL1Y4 118577980 EC50 = 5.4 nM T37693 CY3PA2 118643310 Ki = 78.8 nM T37693 CTC9R6 118643314 Ki = 19.7 nM T37693 C6CG5I 118643315 Ki = 3.3 nM T37693 C3PQS9 118643388 Ki = 360 nM T37693 C6E7PK 118643393 Ki = 8.2 nM T37693 C6XYO1 118643396 Ki = 0.8 nM T37693 CI2AP3 118643406 Ki = 0.7 nM T37693 CIHQ76 118643434 Ki = 750 nM T37693 C7X1ZB 118706308 EC50 = 173.78 nM T37693 CPR53I 118706309 EC50 = 295.12 nM T37693 CC2G6V 118706310 EC50 = 31622.78 nM T37693 C1D2GL 118706311 EC50 = 12589.25 nM T37693 CFL1Z4 118706312 EC50 = 6606.93 nM T37693 C6SD4K 118706313 EC50 = 12022.64 nM T37693 CS79QX 118706314 EC50 = 57543.99 nM T37693 CQ9B4G 118706315 EC50 = 19498.45 nM T37693 C16JGM 118706317 EC50 = 16595.87 nM T37693 CZ24EM 118706318 EC50 = 2884.03 nM T37693 CN4G2U 118707905 Ki = 9180 nM T37693 CUS4F2 118707906 Ki = 22550 nM T37693 CI23QP 118707907 Ki = 1210 nM T37693 C0ABJ8 118709741 Ki = 830 nM T37693 C9AO5K 118709742 Ki = 1890 nM T37693 CF6CR0 118709743 Ki > 10000 nM T37693 C0VP2R 118710167 Ki = 2400 nM T37693 CP7AZ2 118710172 Ki = 12700 nM T37693 CIQ9L8 118710173 Ki = 31000 nM T37693 CSP5J3 118710952 Ki = 119.3 nM T37693 C9CM3X 118710953 Ki = 97.2 nM T37693 CW5S6I 118710954 Ki = 50.2 nM T37693 CW15QT 118710955 Ki = 21.2 nM T37693 CD1A3B 118710956 Ki = 540 nM T37693 CV9Q4L 118710957 Ki = 814.8 nM T37693 CT12DE 118710958 Ki = 230 nM T37693 CE3LG5 118710959 Ki = 2370 nM T37693 CRVG42 118710960 Ki > 10000 nM T37693 CK8C0R 118710961 Ki = 16.4 nM T37693 CCIE15 118710962 Ki = 96.3 nM T37693 C0CS2E 118710963 Ki = 27.9 nM T37693 CJ35MC 118710964 Ki = 202.3 nM T37693 C4WUB9 118710965 Ki > 10000 nM T37693 C37ZAO 118710966 Ki > 10000 nM T37693 C89QBL 118710967 Ki > 10000 nM T37693 CRDH69 118710968 Ki > 10000 nM T37693 C6CP7G 118710969 Ki > 10000 nM T37693 CSE1V9 118710970 Ki = 182.6 nM T37693 CW09BI 118710971 Ki = 677.8 nM T37693 CB8SV3 118710972 Ki = 460 nM T37693 CM91UF 118710973 Ki = 650 nM T37693 C9S5DN 118710974 Ki = 250 nM T37693 CAK1P8 118710975 Ki > 10000 nM T37693 CI9NB6 118710976 Ki = 1520 nM T37693 CYGH30 118710977 Ki = 1850 nM T37693 CJ7UB1 118711121 Ki = 980 nM T37693 CQU6G8 118711283 Ki = 370 nM T37693 CA6F4R 118711284 Ki = 10000 nM T37693 CIH8W4 118712416 Ki > 10000 nM T37693 CD5U3M 118712417 Ki = 4200 nM T37693 CRML68 118712418 Ki = 510 nM T37693 CHD54U 118712419 Ki = 180 nM T37693 COV62X 118712420 Ki = 470 nM T37693 CA3HS1 118712421 Ki = 1000 nM T37693 C4C9AZ 118712672 Ki > 10000 nM T37693 CS76HN 118712673 Ki > 10000 nM T37693 C6F7MO 118716108 IC50 > 10000 nM T37693 CI51GD 118716112 IC50 = 5120 nM T37693 CN4QJ1 118716114 IC50 > 10000 nM T37693 CWL0K7 118716118 IC50 > 10000 nM T37693 CH7C4E 118716121 IC50 > 10000 nM T37693 C9OJX0 118716122 IC50 > 10000 nM T37693 CON02E 118717918 Ki = 0.7943 nM T37693 C3XP4F 118719586 Ki = 3.9 nM T37693 CKXB38 118719587 Ki = 2.82 nM T37693 CVW1U3 118719588 Ki = 2096 nM T37693 C3ZD9J 118719589 Ki = 129 nM T37693 CUF2I9 118719590 EC50 = 23.7 nM T37693 CZDV38 118719591 Ki = 3.6 nM T37693 C46ZPY 118719592 Ki = 18 nM T37693 CO4BY2 118719593 Ki = 176 nM T37693 CJ3N1Q 118719594 Ki = 62.6 nM T37693 CUC56R 118719595 Ki = 27.1 nM T37693 CIAP43 118719596 Ki = 1394 nM T37693 CZJ47G 118719597 Ki = 2466 nM T37693 CWJ26O 118719598 Ki = 1341 nM T37693 CX3UG7 118719599 Ki = 1.36 nM T37693 C8BYZ5 118719600 Ki = 0.56 nM T37693 CXJA89 118719601 Ki = 1.46 nM T37693 C4YA1O 118719602 Ki = 3.83 nM T37693 C40MOC 118719603 Ki = 0.96 nM T37693 CW0L8Y 118719604 Ki = 2.17 nM T37693 C5LA2D 118719605 Ki = 0.27 nM T37693 CPK5M3 118719606 Ki = 0.17 nM T37693 C1NWH9 118719607 Ki = 0.68 nM T37693 C1PD4O 118719608 Ki = 0.35 nM T37693 CRZ25Y 118719763 EC50 > 3000 nM T37693 CMW6F8 118719764 EC50 > 3000 nM T37693 C24QUV 118719765 EC50 > 3000 nM T37693 C9G0VD 118719766 EC50 > 3000 nM T37693 C1UV4W 118719767 EC50 > 3000 nM T37693 C9V5PB 118719768 EC50 > 3000 nM T37693 CRY18I 118719769 EC50 > 3000 nM T37693 CFQ8R2 118719770 EC50 > 3000 nM T37693 CX10UA 118719771 EC50 > 3000 nM T37693 C67DWN 118719772 EC50 > 3000 nM T37693 CK58TI 118719773 EC50 > 3000 nM T37693 CB5NI2 118719774 EC50 > 3000 nM T37693 CK0UW6 118720158 EC50 > 3000 nM T37693 CDW0B1 118720256 EC50 = 41 nM T37693 C05YAJ 118720257 EC50 > 1000 nM T37693 C96TEL 118720552 EC50 = 0.5 nM T37693 C9X6JL 118720553 EC50 = 0.7 nM T37693 CRW5A6 118720554 EC50 = 1.3 nM T37693 C4DJ0Z 118720555 EC50 = 0.2 nM T37693 CSF28U 118720556 EC50 = 3.2 nM T37693 CA2Q0R 118720557 EC50 = 4.2 nM T37693 C17YFC 118720558 EC50 = 21.9 nM T37693 CH0A5R 118720559 EC50 = 1.4 nM T37693 CH0AS9 118720560 EC50 = 5.1 nM T37693 C2AW1O 118720561 EC50 = 5.5 nM T37693 C74UHD 118720562 EC50 = 0.7 nM T37693 CN42VO 118720563 EC50 = 19.8 nM T37693 C6ZT3W 118720564 EC50 = 13.6 nM T37693 CY6T4M 118720565 EC50 = 1.2 nM T37693 CK8V5U 118720566 EC50 = 38.8 nM T37693 C6FDB2 118720567 EC50 = 5.4 nM T37693 CP80QJ 118720568 EC50 = 15.2 nM T37693 CWTU50 118720569 EC50 = 21.2 nM T37693 CI3O6C 118720570 EC50 = 0.4 nM T37693 C6XN4L 118720571 EC50 = 1.1 nM T37693 CDM1K3 118720572 EC50 = 3 nM T37693 CR6VQ9 118720573 EC50 = 38.5 nM T37693 C5OHY6 118720574 EC50 = 100.9 nM T37693 C2TG4E 118720575 EC50 = 19 nM T37693 C42GIB 118720576 EC50 = 7.4 nM T37693 CMIB62 118720577 EC50 = 25.3 nM T37693 C0MXK9 118720578 EC50 = 0.9 nM T37693 CGH7U9 118720579 EC50 = 23000 nM T37693 C9SJH4 118720580 EC50 = 14.6 nM T37693 C0U8PC 118720581 EC50 = 42.4 nM T37693 CRZK09 118720582 EC50 = 809 nM T37693 C62GLY 118720583 EC50 = 25.3 nM T37693 CPB17U 118720584 EC50 = 420.2 nM T37693 C2EDL9 118722126 EC50 = 12.5 nM T37693 CNRL68 118722145 EC50 = 2 nM T37693 CMW3I5 118722146 EC50 = 9.6 nM T37693 CYP8S3 118722147 EC50 = 1.2 nM T37693 C2Q7XA 118722148 EC50 = 37 nM T37693 CY6H0O 118722149 EC50 = 6.2 nM T37693 CW73HU 118722150 EC50 = 6.3 nM T37693 C6GB4N 118722151 EC50 = 32 nM T37693 CVH78O 118722152 EC50 = 73 nM T37693 CCL3B9 118722153 EC50 = 209 nM T37693 CT6J5I 118722154 EC50 = 0.99 nM T37693 CKCR01 118722155 EC50 = 2.6 nM T37693 CZ0R3B 118722156 EC50 = 40 nM T37693 CM3YE9 118722157 EC50 = 12 nM T37693 CLS38E 118722158 EC50 = 7.9 nM T37693 CR2E1P 118722159 EC50 = 56 nM T37693 C4A9RF 118722160 EC50 = 21 nM T37693 CTND40 118722161 EC50 = 14 nM T37693 CBCN25 118722162 EC50 = 47 nM T37693 CS6CX9 118726686 Ki = 2742 nM T37693 C3O6VM 118726687 Ki > 10000 nM T37693 CTW1E4 118726688 Ki = 100 nM T37693 CU2XS4 118726689 Ki = 90 nM T37693 CZS7Q0 118726769 Ki = 60 nM T37693 C2CZ9R 118726770 Ki = 60 nM T37693 C4U0TC 118726771 Ki = 11.48 nM T37693 CBG38P 118726772 Ki = 22 nM T37693 CS91PZ 118727545 Ki > 1000 nM T37693 CK9YC1 118727546 Ki > 1000 nM T37693 CQ1MT5 118727547 Ki > 1000 nM T37693 C6FP4M 118727548 Ki > 1000 nM T37693 CSU24B 118727549 Ki > 1000 nM T37693 CS15CM 118727550 Ki > 1000 nM T37693 CPS6Q0 118728139 EC50 = 1.4 nM T37693 CK18FP 118728140 EC50 > 20 nM T37693 C8CHU4 118728141 EC50 > 20 nM T37693 CV8YP1 118728142 EC50 = 5 nM T37693 CBDX93 118731518 Ki = 0.7 nM T37693 C7CIR8 118731519 Ki = 3.9 nM T37693 CPY68L 118732562 EC50 = 972 nM T37693 CWYR05 118732564 EC50 = 130 nM T37693 C5BUD9 118732565 EC50 = 321 nM T37693 C5OD3H 118732567 IC50 > 10000 nM T37693 CXI3Y5 118732568 IC50 > 10000 nM T37693 C7HPJ3 118732569 IC50 = 22 nM T37693 C3FXW5 118732570 IC50 = 1177 nM T37693 CV52GQ 118732571 IC50 = 162 nM T37693 CY31XU 118732572 IC50 = 28 nM T37693 C12WUS 118732573 IC50 = 20 nM T37693 CBL75P 118732574 IC50 = 19 nM T37693 CUMB75 118732575 Ki = 0.0869 nM T37693 C4VYR9 118732586 Ki = 43.95 nM T37693 CTUA83 118733872 Ki > 1000 nM T37693 CME84I 118733873 Ki = 337 nM T37693 CA60FT 118733874 Ki = 8.4 nM T37693 CNJ46O 118733875 Ki = 4.2 nM T37693 C1WE6Z 118733876 Ki > 1000 nM T37693 CU41FJ 118733877 Ki = 13.1 nM T37693 C0JPQ1 118733878 Ki = 24.8 nM T37693 C5V2QA 118733879 Ki = 4.6 nM T37693 CDO6G2 118733880 Ki > 1000 nM T37693 CY80VZ 118733881 Ki = 10.3 nM T37693 C6UY8Q 118733882 Ki = 9.6 nM T37693 C2MHZ6 118734857 Ki = 398 nM T37693 C1IEC4 118734858 Ki = 597 nM T37693 CA6R8C 118735104 Ki > 3000 nM T37693 CZK9S4 118735105 Ki > 3000 nM T37693 C9VBC6 118735106 Ki > 3000 nM T37693 CCZ36J 118735107 Ki > 3000 nM T37693 CH1N5T 118735108 Ki > 3000 nM T37693 CFLH28 118735109 Ki = 29.2 nM T37693 C6BTX2 118735110 Ki > 3000 nM T37693 CNUC23 118735111 Ki > 3000 nM T37693 CV0RP2 118735112 Ki > 3000 nM T37693 CP21CI 118735884 Ki = 0.75 nM T37693 C14OKB 118735885 Ki = 4.2 nM T37693 C5T2XB 118735886 Ki = 25.4 nM T37693 C89UAT 118735887 Ki = 19.8 nM T37693 C58TLB 118735888 Ki = 1.5 nM T37693 CB9CH4 118735889 Ki = 36 nM T37693 CTC74N 118735890 Ki = 0.75 nM T37693 CK38BW 118735891 Ki = 7.44 nM T37693 CG6XJ8 118735892 Ki = 11.2 nM T37693 CPA03J 118735893 Ki = 215 nM T37693 CX4PY8 121028259 EC50 > 10000 nM T37693 CN8T4V 121283196 Ki = 1.2 nM T37693 CYJ30U 121283240 Ki = 7.1 nM T37693 C4K1LD 122179273 EC50 = 154.8 nM T37693 CYC52P 122179274 EC50 = 4007.5 nM T37693 CXJU68 122179275 EC50 = 27 nM T37693 C45ZET 122179276 EC50 = 396.1 nM T37693 C3KL4C 122179277 Ki = 3958.3 nM T37693 CBT8V5 122179278 Ki > 10000 nM T37693 CZ3NY8 122179279 EC50 = 2.9 nM T37693 C3A0JR 122179280 EC50 = 9.6 nM T37693 CUTL72 122179281 Ki = 2.5 nM T37693 C9QHM7 122180086 Ki = 129 nM T37693 CCY7M4 122180087 Ki = 335 nM T37693 C8Z6KE 122180088 Ki = 912 nM T37693 C1MY7T 122182962 Ki > 10000 nM T37693 CX0D8H 122182963 IC50 > 10000 nM T37693 CM9Z1Y 122182964 Ki > 10000 nM T37693 CTF89J 122182965 Ki > 10000 nM T37693 CL7FR1 122182966 Ki > 10000 nM T37693 CDUA90 122182967 Ki > 10000 nM T37693 CB3V2C 122182968 Ki > 10000 nM T37693 CN5H3A 122182969 Ki > 10000 nM T37693 C4HI6P 122182970 Ki > 10000 nM T37693 C9QDS4 122182971 Ki > 10000 nM T37693 C5CL4O 122182972 IC50 > 10000 nM T37693 C1SVF8 122182973 Ki > 10000 nM T37693 CP8GV4 122182974 Ki > 10000 nM T37693 C9QMW0 122182975 Ki > 10000 nM T37693 C3I7FO 122182976 IC50 > 10000 nM T37693 CXR07B 122183469 Ki = 1030 nM T37693 CWP92F 122183470 Ki = 860 nM T37693 CO2P0J 122186206 Ki > 10000 nM T37693 CVA4X9 122186207 Ki = 1589 nM T37693 CIMB95 122186208 EC50 = 118 nM T37693 C9M4RG 122186209 Ki = 2618 nM T37693 C6T7FD 122186210 Ki > 10000 nM T37693 C21IXD 122186211 EC50 > 5000 nM T37693 CI39PN 122186212 Ki > 10000 nM T37693 C1JKN9 122186213 EC50 = 29.5 nM T37693 CLYT85 122186214 Ki = 1717 nM T37693 C8SK3V 122186215 EC50 = 28.8 nM T37693 C3I6RX 122186216 Ki = 160.7 nM T37693 C42KBM 122186217 EC50 = 254 nM T37693 CI0S8P 122186218 Ki = 3166 nM T37693 CPLO68 122186219 EC50 > 5000 nM T37693 CL91KO 122186220 EC50 = 89.7 nM T37693 C0B9OG 122186221 EC50 > 5000 nM T37693 CEPZ53 122186222 EC50 > 5000 nM T37693 CLXN43 122186223 EC50 > 5000 nM T37693 C4FA8H 122186224 Ki > 10000 nM T37693 CM1HG9 122186225 Ki > 10000 nM T37693 CYE3S0 122186226 Ki > 10000 nM T37693 CL7QJ3 122188721 Ki = 5.7 nM T37693 C6LEJ5 122188722 Ki = 343 nM T37693 C0Y7MH 122188723 Ki = 164 nM T37693 C1LKQ8 122188724 Ki > 5000 nM T37693 CL6ZK9 122188725 Ki = 72.2 nM T37693 CY8A0I 122188726 Ki > 5000 nM T37693 CNOJ38 122188727 Ki > 5000 nM T37693 CM12WF 122188728 Ki = 1100 nM T37693 CZ5K3W 122188729 Ki > 5000 nM T37693 C03CJH 122188730 Ki = 492 nM T37693 CN36ST 122188731 Ki = 244 nM T37693 C0Y2HU 122188732 Ki = 106 nM T37693 CY89ZL 122188733 Ki = 1707 nM T37693 CG8AB5 122188734 Ki > 5000 nM T37693 CASB97 122188735 Ki > 5000 nM T37693 C46EAN 122188736 Ki = 575 nM T37693 CKPT42 122188737 Ki > 5000 nM T37693 C5SNP3 122188738 Ki > 5000 nM T37693 C5HC0Z 122188739 Ki > 5000 nM T37693 CPE05A 122188740 Ki = 343 nM T37693 CB5NH1 122188741 Ki = 7.2 nM T37693 CDA10L 122366667 Ki = 2220 nM T37693 C16IOX 123128346 IC50 > 10000 nM T37693 C3DWH0 123627357 EC50 = 1.2 nM T37693 CUW54Z 123922722 EC50 = 560 nM T37693 CDK95B 124021285 EC50 = 3.8 nM T37693 CCQO62 126630141 EC50 = 7400 nM T37693 CZ6G3E 126630168 EC50 = 5900 nM T37693 C8CBI0 127026099 Ki = 1545 nM T37693 CGFD26 127027049 Ki = 1041 nM T37693 CYN8P2 127027323 Ki = 1785 nM T37693 CIR76K 127027671 Ki = 4407 nM T37693 C6E1TL 127027672 Ki = 4719 nM T37693 CXK8J7 127027699 Ki = 1808 nM T37693 CED8I2 127027701 Ki = 2496 nM T37693 CO32AZ 127027987 Ki = 6213 nM T37693 CM8VA4 127027989 Ki > 20000 nM T37693 C4BY3G 127028018 Ki = 1725 nM T37693 C18JNK 127029837 Ki = 523 nM T37693 CZX4C2 127029838 Ki = 6392 nM T37693 C9FG1J 127029891 Ki = 53 nM T37693 CT81PH 127029928 Ki = 825 nM T37693 C39OXL 127029929 Ki = 509 nM T37693 CY3LI1 127029930 Ki = 6 nM T37693 C5SH7V 127030115 Ki > 10000 nM T37693 CN49LK 127030116 IC50 = 26.9 nM T37693 CV6Z5S 127030117 Ki = 4 nM T37693 C1U2CM 127030118 Ki = 198 nM T37693 C3L8GO 127030160 Ki > 40000 nM T37693 C3I4CH 127030161 Ki = 1073 nM T37693 CHMI58 127030184 Ki = 69.43 nM T37693 CVDP63 127030185 Ki = 143 nM T37693 CMO64X 127030260 Ki = 5517 nM T37693 CYBU18 127030261 Ki > 40000 nM T37693 C61MQJ 127030421 Ki > 10000 nM T37693 CN7A6R 127030422 Ki > 40000 nM T37693 CIMH58 127030534 Ki = 25 nM T37693 CXBY26 127030535 Ki = 674 nM T37693 CLRC71 127030536 Ki = 383 nM T37693 C4HSR6 127030537 Ki = 43 nM T37693 C2NVB3 127030843 Ki = 514 nM T37693 C4WXA8 127030844 Ki = 48 nM T37693 C9F2UM 127030845 Ki = 8.4 nM T37693 C3Y6ZT 127031443 Ki = 47 nM T37693 CTE32L 127031950 Ki = 152 nM T37693 CM7DG0 127032456 IC50 > 10000 nM T37693 CBE3R6 127032540 Ki = 414 nM T37693 C7L8BN 127032985 Ki = 6.8 nM T37693 CA7HV0 127032986 Ki = 45 nM T37693 C3YG8K 127033294 Ki = 228 nM T37693 CUNJ13 127033295 Ki = 716 nM T37693 C6JM5H 127033296 Ki > 10000 nM T37693 CSGK03 127033297 Ki > 10000 nM T37693 CZ73AN 127033298 Ki = 982 nM T37693 CL47YF 127033299 Ki = 1332 nM T37693 C6XWZ5 127033300 Ki = 21 nM T37693 CDFJ81 127033483 Ki = 4923 nM T37693 C2L0UO 127033585 Ki = 1352 nM T37693 C5WK8C 127033586 Ki = 158 nM T37693 CXG07N 127033786 Ki = 1578 nM T37693 C8N0RD 127033787 Ki > 40000 nM T37693 CB9OZ6 127034064 Ki > 40000 nM T37693 C9D8NR 127034065 Ki > 40000 nM T37693 C30BCV 127034066 Ki > 40000 nM T37693 CK57OG 127034067 Ki > 40000 nM T37693 CEH0S2 127034069 Ki = 698 nM T37693 CSK5Y7 127034071 Ki = 3604 nM T37693 C6GPQ0 127034073 Ki = 15.4 nM T37693 C0KBT1 127034080 Ki > 40000 nM T37693 CQ9N4O 127034141 Ki = 117 nM T37693 COA3U0 127034142 Ki = 11.3 nM T37693 CST04W 127034143 Ki = 96 nM T37693 CP43EW 127034294 IC50 = 3.5 nM T37693 CD4VN6 127034337 Ki = 515 nM T37693 C56NPM 127034412 Ki = 47 nM T37693 CE7U2X 127034413 Ki = 31 nM T37693 C75HWE 127034414 Ki = 22 nM T37693 CE51CW 127034415 Ki = 566 nM T37693 CL4DX7 127034588 EC50 = 2.6 nM T37693 C7LXG3 127045805 Ki >= 10000 nM T37693 CX40GI 127045919 Ki = 594 nM T37693 CQ56AZ 127045920 Ki = 2667 nM T37693 C6AC8U 127046131 Ki = 196 nM T37693 CQ0FN3 127046132 Ki = 337 nM T37693 C5JV3I 127046164 Ki = 1783 nM T37693 C6WYM3 127046377 Ki > 10000 nM T37693 C7D9MJ 127046378 Ki > 10000 nM T37693 C4QH0N 127046416 Ki = 265 nM T37693 C5XD4U 127046684 Ki = 166 nM T37693 C2BP4Q 127046685 Ki = 1413 nM T37693 C9PW8O 127046686 Ki = 84.1 nM T37693 CCU7A4 127046687 Ki = 1106 nM T37693 COLP16 127047329 Ki = 103 nM T37693 CGV6Y5 127047410 Ki = 352 nM T37693 CY80XQ 127047411 Ki = 1262 nM T37693 CXD79Z 128708882 EC50 = 290 nM T37693 C5BLU7 128939360 IC50 = 6500 nM T37693 CO0WB4 129257195 Ki = 1.2 nM T37693 CL2A1B 129781980 Ki = 1600 nM T37693 C8D3MY 130366796 Ki > 10000 nM T37693 CJHT67 132510986 IC50 = 4.2 nM T37693 CB1D8Q 132578438 Ki = 53 nM T37693 C50HGD 132578440 Ki = 33 nM T37693 C2AKW3 132585222 EC50 = 13.99 nM T37693 CNSG54 132585223 EC50 = 48.74 nM T37693 CDK60Q 134130813 Ki = 1000 nM T37693 CDP7U0 134131733 Ki = 300 nM T37693 C1Q9XZ 134131985 Ki > 10000 nM T37693 CF64DG 134132091 EC50 = 4660 nM T37693 CLR9C6 134132855 Ki = 300 nM T37693 C7B4JU 134133334 Ki = 540.1 nM T37693 CWG8P2 134133524 Ki = 900 nM T37693 CTI0Y2 134133618 Ki = 600 nM T37693 CFTS48 134134129 EC50 = 1450 nM T37693 CV8SR9 134134298 Ki = 80 nM T37693 C7IEV8 134135104 EC50 > 10000 nM T37693 C4ILM0 134135334 Ki = 1600 nM T37693 C7BQ5W 134135465 EC50 > 10000 nM T37693 C5WFH6 134135522 EC50 = 743 nM T37693 COI6K4 134135649 Ki = 1900 nM T37693 CK0RA6 134135962 Ki = 170.81 nM T37693 C3K9NQ 134136117 EC50 > 10000 nM T37693 C4NBF7 134136193 EC50 = 370 nM T37693 C1ZW2U 134136510 Ki = 800 nM T37693 C5JQ6R 134136907 EC50 > 11000 nM T37693 C9J5KY 134137187 Ki = 100 nM T37693 CUG02L 134137271 Ki = 300 nM T37693 C32UGQ 134137479 Ki = 584.17 nM T37693 CY2EK1 134137727 Ki = 500 nM T37693 C3Y6FA 134138389 EC50 = 1760 nM T37693 C0OHC7 134138469 EC50 = 1610 nM T37693 C3J6GU 134138518 EC50 > 10000 nM T37693 CW1KO0 134138598 Ki > 10000 nM T37693 CIM01Y 134138796 EC50 > 10000 nM T37693 C7T2EY 134138952 EC50 > 10000 nM T37693 CTZ5Q6 134139255 EC50 = 3240 nM T37693 CGTZ26 134139273 EC50 = 2910 nM T37693 C1NJ9C 134139421 Ki = 400 nM T37693 CJ1FG3 134139799 Ki = 58.28 nM T37693 C4Z0KB 134140018 Ki = 700 nM T37693 CDB9F4 134140655 EC50 > 10000 nM T37693 C2QGM7 134140841 EC50 = 2000 nM T37693 C1HD0Q 134140959 EC50 = 807 nM T37693 C6GJB1 134141428 Ki > 10000 nM T37693 CTZ4H5 134141506 Ki = 1500 nM T37693 C95QFU 134141929 EC50 = 650 nM T37693 CZ3H1I 134142321 Ki = 700 nM T37693 CC4H7W 134142473 Ki = 700 nM T37693 CITW76 134142657 EC50 = 560 nM T37693 CW4N6H 134142675 EC50 > 10000 nM T37693 C5Y9UW 134142847 Ki = 1400 nM T37693 CGN42L 134143149 EC50 = 7850 nM T37693 C2M9IN 134143205 EC50 > 10000 nM T37693 CNT6D2 134143262 Ki = 500 nM T37693 CVT6D2 134144382 Ki > 10000 nM T37693 CNF1C8 134144706 Ki = 57 nM T37693 CL8T0G 134145050 EC50 > 10000 nM T37693 CN7TR5 134145283 EC50 > 10000 nM T37693 C4S2FX 134146248 Ki = 300 nM T37693 C3E4RW 134146777 EC50 = 8610 nM T37693 CP82DL 134146936 EC50 = 1940 nM T37693 CWV4H0 134147498 Ki = 52.1 nM T37693 C84IHR 134148177 Ki = 500 nM T37693 CERX86 134148188 EC50 = 1270 nM T37693 CUV40N 134148570 Ki = 718.2 nM T37693 C89YTJ 134149018 Ki > 10000 nM T37693 CR64GQ 134149040 Ki > 10000 nM T37693 C07FSW 134149771 Ki = 400 nM T37693 CH9DW2 134149775 EC50 > 10000 nM T37693 CBF56O 134149796 EC50 = 1130 nM T37693 C1W4ID 134149884 EC50 = 9410 nM T37693 C97HGO 134150139 Ki = 167.81 nM T37693 C5IXY8 134150287 Ki = 546.44 nM T37693 C5YG9D 134150307 EC50 > 10000 nM T37693 C7TJY0 134150441 Ki = 84.22 nM T37693 CU63GK 134151463 EC50 > 10000 nM T37693 CPZR93 134152278 EC50 > 10000 nM T37693 CHA9B0 134152389 EC50 > 10000 nM T37693 C8NGJ4 134152497 EC50 = 854 nM T37693 CG6M0R 134152684 EC50 = 3660 nM T37693 CED06W 134154057 Ki > 10000 nM T37693 CJX45N 134154719 EC50 > 10000 nM T37693 CC5TU4 134154932 EC50 > 10000 nM T37693 CZOY08 134155237 EC50 > 10000 nM T37693 C0MVG7 134155406 Ki = 6.15 nM T37693 CJ1BA3 134155808 EC50 > 10000 nM T37693 CML28S 134155966 Ki = 100 nM T37693 C8QIC2 134156159 EC50 = 1310 nM T37693 C0M2GZ 134156537 Ki > 10000 nM T37693 C6KS0N 134156578 Ki = 1900 nM T37693 C92VRD 134156729 Ki = 20.02 nM T37693 CEW50T 134156883 EC50 = 3820 nM T37693 CYCE87 134157291 Ki = 800 nM T37693 C0JL7I 134157399 EC50 = 5550 nM T37693 CYS3B9 134157891 EC50 > 10000 nM T37693 CNX5J2 134157932 Ki = 7.59 nM T37693 CNDI28 135156076 Ki = 110 nM T37693 CK8T9E 135156097 Ki = 630 nM T37693 CX2SZ4 135156106 Ki > 10000 nM T37693 C1W9FV 135156138 Ki = 3200 nM T37693 C7UJ0A 135156140 Ki = 4600 nM T37693 CIS28F 135156142 Ki > 10000 nM T37693 C7B0UK 135156143 Ki = 1300 nM T37693 CN83XY 135156151 Ki > 10000 nM T37693 CWEU47 135156153 Ki = 2100 nM T37693 COC48A 135156160 Ki = 6500 nM T37693 CGBP75 135156161 Ki = 990 nM T37693 CYE13V 135156182 Ki > 10000 nM T37693 C0BLS7 135156185 Ki > 10000 nM T37693 CF29ML 135156190 Ki = 8500 nM T37693 CWU6L2 135156193 Ki = 620 nM T37693 CS9RP5 135156203 Ki = 740 nM T37693 CLS4A8 135156215 Ki > 10000 nM T37693 CUI9X6 135156216 Ki > 10000 nM T37693 CED38C 135156219 Ki = 3600 nM T37693 C8BZ2J 135156223 Ki = 850 nM T37693 C0UO9X 135156228 Ki = 1700 nM T37693 C4K1NW 135156229 Ki = 420 nM T37693 CXV38J 135156232 Ki = 2300 nM T37693 CM4LS9 135156237 Ki > 10000 nM T37693 C5U9ZM 135156239 Ki > 10000 nM T37693 CA82SP 135156240 Ki = 980 nM T37693 CY8D4L 135156241 Ki = 500 nM T37693 CJ85SW 135156242 Ki = 5100 nM T37693 C1GY2T 135156251 EC50 > 10000 nM T37693 CINV95 135156278 Ki > 10000 nM T37693 C4C8FY 135156279 Ki > 10000 nM T37693 CX8JS3 135156281 Ki = 7100 nM T37693 C3AYS7 135156282 Ki = 400 nM T37693 C4Y3XH 135156284 Ki > 10000 nM T37693 CQW0X9 135156285 Ki = 2400 nM T37693 COW34N 135156292 Ki > 10000 nM T37693 CR4A9I 135156296 Ki = 4200 nM T37693 CK2C8T 135156317 Ki > 10000 nM T37693 C5VA0M 135156319 Ki > 10000 nM T37693 C0GE5U 135156322 Ki > 10000 nM T37693 C1NX8O 135156329 Ki = 2000 nM T37693 C5YP0R 135156335 Ki = 130 nM T37693 CSX16V 135156341 Ki > 10000 nM T37693 CUE5F7 135156347 Ki = 740 nM T37693 CXT1L3 135156354 Ki = 610 nM T37693 CL6P8W 135156382 Ki = 9000 nM T37693 CNW3I9 135156391 Ki = 5000 nM T37693 CR29YT 135156426 Ki > 10000 nM T37693 CN2RT9 135156435 Ki > 10000 nM T37693 CDY28G 135156437 Ki > 10000 nM T37693 C6L3MW 135156439 Ki = 2800 nM T37693 CFU36D 135156440 Ki > 10000 nM T37693 CQ7O9J 135156442 Ki > 10000 nM T37693 C2HPY7 135156445 Ki > 10000 nM T37693 CR1Z4C 135156452 Ki = 860 nM T37693 C7L6QM 135156454 Ki > 6000 nM T37693 CNMF20 135156469 Ki = 2300 nM T37693 CBSC28 135156470 Ki > 10000 nM T37693 C7YIQ0 135156473 Ki = 1700 nM T37693 CYML32 135156477 Ki > 10000 nM T37693 C25ENA 135156501 Ki > 10000 nM T37693 C3NQ7M 135156503 Ki = 1300 nM T37693 CBV81U 135156509 Ki > 10000 nM T37693 CVW76H 135156513 Ki = 1400 nM T37693 CJM59S 135164381 Ki = 3400 nM T37693 C80TDY 135164613 Ki = 2700 nM T37693 C92DIW 135165004 Ki > 6000 nM T37693 C19PYU 135165007 Ki > 10000 nM T37693 C3ROX7 135376339 IC50 > 10000 nM T37693 CY9M3O 135376387 IC50 = 3400 nM T37693 CA3S6K 135376388 IC50 > 10000 nM T37693 C3XV6H 135376400 IC50 = 4100 nM T37693 CZ10DT 135376603 IC50 > 10000 nM T37693 CD3V1F 135376751 IC50 > 10000 nM T37693 C3L8EB 135881473 EC50 = 84 nM T37693 CH31WM 135881474 EC50 = 645.5 nM T37693 CTA68K 135881483 Ki = 13.9 nM T37693 C0R5SW 135881484 EC50 = 143.4 nM T37693 CSB01I 135881485 EC50 = 9.8 nM T37693 CZJ2F3 135881488 EC50 = 186.9 nM T37693 C5CWR3 135881490 Ki = 58.8 nM T37693 C07DOW 135881494 EC50 = 79.1 nM T37693 C43MYR 135881498 EC50 = 202.2 nM T37693 CRQ1H4 135922724 IC50 > 10000 nM T37693 C8UG5X 135922725 IC50 > 10000 nM T37693 CI86RJ 135923581 IC50 = 7300 nM T37693 C04MQH 135923694 IC50 = 8600 nM T37693 C8DOW1 135923695 IC50 = 5500 nM T37693 CUQC19 135923696 IC50 > 2000 nM T37693 CO3SU7 135924633 EC50 = 88.2 nM T37693 C28CMN 135924634 EC50 = 5.8 nM T37693 CF17PG 135924635 EC50 = 85 nM T37693 C1Y6IV 135924636 EC50 = 18 nM T37693 CQFV38 135924637 EC50 = 102 nM T37693 CWH7R6 135924638 EC50 = 540 nM T37693 CH5MI8 135924639 EC50 = 492 nM T37693 CO2FL0 135924640 EC50 = 28.7 nM T37693 C0OP6U 135924641 EC50 = 14.7 nM T37693 C2XBO9 135924642 EC50 = 15.9 nM T37693 CIGQ76 135924643 EC50 = 11.7 nM T37693 CH37QR 135924644 EC50 = 43 nM T37693 C8F4SQ 135924645 EC50 = 13.3 nM T37693 CI4SU6 135924646 EC50 = 10 nM T37693 CDL89Z 135924647 EC50 = 71.6 nM T37693 C04MZE 135930698 EC50 = 188.7 nM T37693 C9ROE1 135936176 Ki > 40000 nM T37693 CE26DH 135936177 Ki > 40000 nM T37693 C0WB3A 135936178 Ki > 40000 nM T37693 CXH73Y 135936179 Ki > 40000 nM T37693 CCOB67 135936180 Ki = 270 nM T37693 CD3K1W 135936181 Ki > 40000 nM T37693 CAX5E8 135981703 Ki = 387 nM T37693 CSRK39 135995913 EC50 = 92.68 nM T37693 C8S1ME 135995914 EC50 = 496.59 nM T37693 CI7Z5E 135995915 EC50 = 17900 nM T37693 C2RG1O 135995916 EC50 > 10000 nM T37693 CVZ6G2 135995917 EC50 = 341 nM T37693 C0RH1T 135995918 EC50 = 472 nM T37693 C31RKJ 135995919 EC50 = 1580 nM T37693 C0DQ2F 135995920 EC50 > 10000 nM T37693 C1APX3 135995921 EC50 = 476.43 nM T37693 CTG9L5 135995922 EC50 = 993 nM T37693 C5O9AI 135995923 EC50 = 219.79 nM T37693 CNHL53 135995924 EC50 = 127 nM T37693 C36XJL 135995925 EC50 = 503 nM T37693 CG7C6Z 135995926 EC50 = 57.94 nM T37693 COR21T 135995927 EC50 = 2387.81 nM T37693 CXC32Y 135995928 EC50 > 10000 nM T37693 C39DSU 135995929 EC50 > 10000 nM T37693 C3TWF4 135995930 EC50 > 10000 nM T37693 CA6RF7 135995931 EC50 = 316.96 nM T37693 C0LJQ3 135995932 EC50 > 10000 nM T37693 C74RUI 135995933 EC50 > 10000 nM T37693 CXF8I9 135995934 EC50 = 1415.79 nM T37693 C0W6AO 135995935 EC50 > 10000 nM T37693 C86KWU 135995936 EC50 = 797 nM T37693 C5TOD3 135995937 EC50 = 748.17 nM T37693 CDL8C1 135995938 EC50 = 669.88 nM T37693 C5TF8G 135995939 EC50 = 319.89 nM T37693 C2E5KG 135995940 EC50 = 75.3 nM T37693 CDQ54M 135995941 EC50 = 103.99 nM T37693 CNC8O4 135995942 EC50 = 36.3 nM T37693 CA8QI4 135995943 IC50 = 9.03 nM T37693 C30QJD 135995944 IC50 = 194 nM T37693 CT3DY8 135995945 IC50 > 10000 nM T37693 CTX8Y4 135995946 IC50 = 93.3 nM T37693 CG8H3C 135995947 IC50 = 1480 nM T37693 CJ4W5Y 135995948 IC50 > 10000 nM T37693 C4AQC1 135995949 IC50 = 81.7 nM T37693 C9JBO5 135995950 IC50 = 957 nM T37693 C42UVC 135995951 IC50 = 45.3 nM T37693 CQFZ04 136059727 IC50 > 2000 nM T37693 CW0OS1 136266294 IC50 = 4190 nM T37693 C86HUN 136266296 IC50 > 10000 nM T37693 CV9J6O 136266306 IC50 > 10000 nM T37693 C8EIW4 136266307 IC50 = 1510 nM T37693 CP17HJ 136266308 IC50 = 1680 nM T37693 C1M7XU 136266314 IC50 > 10000 nM T37693 CGE38A 136266318 IC50 = 1650 nM T37693 C7AU4T 136266319 EC50 > 10000 nM T37693 C5EB1A 136266320 EC50 > 10000 nM T37693 CNAG68 136266324 EC50 = 43.95 nM T37693 CD75IA 136266326 IC50 > 10000 nM T37693 C7SGJ1 136266328 IC50 > 10000 nM T37693 CNT63W 137062188 EC50 = 74.99 nM T37693 CD7B2E 137062189 EC50 = 111.94 nM T37693 CIP3Z7 137062190 EC50 = 115.88 nM T37693 C3A0PC 137062191 EC50 = 82.7 nM T37693 C43HNY 137062192 EC50 = 41.02 nM T37693 C40YWC 137062193 EC50 = 20 nM T37693 C9G4KR 137062194 EC50 = 90.7 nM T37693 CPW0D2 137346241 IC50 = 260 nM T37693 C61JRN 137346243 IC50 = 12 nM T37693 CE9HS4 137346244 EC50 = 32 nM T37693 C45CDW 137631524 EC50 = 160 nM T37693 C0BQ4E 137632278 EC50 = 29 nM T37693 C9E1NY 137632735 EC50 = 430 nM T37693 C92XMB 137632971 EC50 = 68.33 nM T37693 CH0B6U 137634141 EC50 = 147.4 nM T37693 CEX02D 137634149 EC50 = 370.2 nM T37693 CY5UW7 137634172 Ki = 2.6 nM T37693 CMR71I 137634355 EC50 = 180 nM T37693 CRA1X6 137634457 Ki = 311 nM T37693 C3CT4W 137635042 EC50 = 113.3 nM T37693 C28BRS 137635194 EC50 = 180 nM T37693 CV97TL 137635223 EC50 = 722.1 nM T37693 CF13WZ 137635764 EC50 > 10000 nM T37693 C9GA2C 137635913 Ki = 763.6 nM T37693 C3Y1MV 137636504 EC50 = 8600 nM T37693 CI5B1C 137636709 EC50 = 308.8 nM T37693 CMWF74 137637124 Ki = 4700 nM T37693 CR7N8A 137637773 EC50 > 10000 nM T37693 CEW9I5 137637866 EC50 = 140 nM T37693 C4IC9D 137637998 EC50 = 23.53 nM T37693 CDZW38 137638255 Ki = 4.4 nM T37693 CHK9C2 137638966 EC50 = 610 nM T37693 CG16DR 137638994 Ki > 1000 nM T37693 C5A7DC 137639252 EC50 = 111.9 nM T37693 C8XHT3 137639360 Ki = 4.9 nM T37693 C5HV6S 137639623 EC50 = 178.2 nM T37693 C2GEU5 137639906 Ki > 1000 nM T37693 CME1D4 137640026 EC50 > 10000 nM T37693 CCY7B8 137640363 Ki > 1000 nM T37693 CAE30M 137640406 IC50 = 19952.62 nM T37693 C8HGN7 137640596 EC50 = 160 nM T37693 C1M7NV 137640777 EC50 = 59 nM T37693 C4TUW2 137640869 EC50 > 10000 nM T37693 CUE37K 137641100 EC50 = 38.22 nM T37693 C3MTB4 137641509 EC50 = 7130 nM T37693 CTR8E0 137641522 Ki = 1900 nM T37693 C98FBN 137642085 Ki = 2 nM T37693 CEYG80 137642209 Ki > 1000 nM T37693 CH80BJ 137643152 EC50 = 394.9 nM T37693 CCBH92 137643269 EC50 = 52.71 nM T37693 CWA3I4 137643432 EC50 = 213.7 nM T37693 CI6NL3 137643518 Ki > 4000 nM T37693 CE6C5S 137643758 EC50 = 410 nM T37693 CXER43 137644281 EC50 > 10000 nM T37693 CLN0W5 137644328 Ki = 7.6 nM T37693 C5YX8V 137644344 IC50 = 16 nM T37693 CR25ML 137644618 EC50 = 31 nM T37693 C3WG9A 137645129 EC50 = 200 nM T37693 CAN3G2 137645158 Ki = 4.7 nM T37693 C1DHM4 137645326 Ki = 1000 nM T37693 C9WC1Z 137645377 EC50 = 40 nM T37693 CNGB09 137645429 EC50 = 78.59 nM T37693 C24LWN 137646015 EC50 = 92 nM T37693 CP9LT8 137647595 EC50 = 226.8 nM T37693 CETC84 137647970 EC50 = 86.51 nM T37693 C7AR3I 137648068 EC50 = 75 nM T37693 C68HNE 137648160 EC50 = 766.8 nM T37693 CBPK31 137648694 Ki = 4800 nM T37693 C5M2VE 137648805 Ki = 4.3 nM T37693 C26JNU 137649145 EC50 > 10000 nM T37693 CVF9U7 137649354 EC50 = 38 nM T37693 CY0WQ7 137649436 IC50 = 7943.28 nM T37693 C9OYR4 137650162 EC50 = 1250 nM T37693 C4QFY0 137650412 EC50 = 99.57 nM T37693 CH50RP 137650702 Ki = 14400 nM T37693 C7NCY0 137650808 EC50 = 100 nM T37693 C2AS9T 137650812 EC50 = 62 nM T37693 CK7RD3 137650977 Ki = 44 nM T37693 CWZ92Q 137651267 IC50 > 10000 nM T37693 CZ2G6N 137651928 EC50 = 490 nM T37693 C0LI1Q 137652040 Ki = 353.4 nM T37693 CBLJ46 137652132 EC50 = 150 nM T37693 C6OZG5 137652212 EC50 = 420 nM T37693 CAS6R5 137652818 EC50 = 3800 nM T37693 C3WI7F 137652938 EC50 = 743.2 nM T37693 CIJW29 137653436 EC50 = 1420 nM T37693 CS13JP 137654029 Ki = 5.7 nM T37693 CCJ74L 137654157 EC50 > 10000 nM T37693 CI18ZR 137654462 EC50 = 27.69 nM T37693 C0C5OB 137654571 Ki = 10400 nM T37693 CPS17B 137654744 EC50 > 10000 nM T37693 C02YDQ 137655423 Ki = 240 nM T37693 C10OJC 137655779 EC50 > 10000 nM T37693 C4HA0W 137655793 Ki = 3.4 nM T37693 C3P0YS 137655815 EC50 = 46.79 nM T37693 CQ6WP9 137656152 EC50 = 720 nM T37693 CWOP62 137657204 EC50 = 82 nM T37693 CE86PO 137657290 EC50 = 85 nM T37693 C6GBO0 137657351 EC50 = 467.6 nM T37693 C1NE5M 137658020 Ki = 961.8 nM T37693 CE5ZL4 137658307 IC50 = 28 nM T37693 CQC6G7 137658542 Ki = 384.5 nM T37693 C6UGE2 137658648 Ki = 426 nM T37693 C5LC2S 137658778 Ki = 13 nM T37693 CG5BW8 137658946 Ki = 16 nM T37693 C8E1VH 137659045 IC50 = 3981.07 nM T37693 CO1SG5 137659148 EC50 = 406.9 nM T37693 C9NT8H 137659169 EC50 = 220 nM T37693 CHOV65 137659408 EC50 = 500 nM T37693 CZ2W6A 137659657 EC50 = 410 nM T37693 CEB89F 137659726 EC50 = 270 nM T37693 CKN42C 137660440 EC50 = 410 nM T37693 CK0AC9 137660701 Ki = 3.3 nM T37693 CY93TX 137661282 EC50 > 10000 nM T37693 CXC4M7 137661310 EC50 = 120 nM T37693 C49PIC 137661579 EC50 = 4700 nM T37693 CP5QB4 137662088 EC50 = 269.5 nM T37693 CB8IM1 138319671 IC50 > 10000 nM T37693 C4SY8V 138491556 EC50 = 0.46 nM T37693 C82LVN 138491578 EC50 = 0.08 nM T37693 CZQ61R 138491579 EC50 = 7.3 nM T37693 CA07WZ 141463725 EC50 = 47.68 nM T37693 C2XU4C 141463726 EC50 = 96.24 nM T37693 CPZ62D 141463727 EC50 > 10000 nM T37693 CYU0K3 141463728 EC50 = 349 nM T37693 CINT06 141463729 EC50 = 594 nM T37693 C2FMK0 141463730 EC50 = 3.665 nM T37693 C7I8XT 141463734 EC50 = 3453 nM T37693 C93LEZ 141463736 EC50 = 34.42 nM T37693 CHDV64 141463737 EC50 > 10000 nM T37693 CTGM15 141463743 EC50 = 396.2 nM T37693 CJA91I 141463744 EC50 = 18.08 nM T37693 C1MSD2 141463745 EC50 = 398.2 nM T37693 CXY8V2 141463746 EC50 = 49.35 nM T37693 CET5X6 141463751 EC50 = 841.9 nM T37693 CYI8H5 141463752 EC50 = 8425 nM T37693 C4F7KJ 141463753 EC50 = 4.955 nM T37693 CGL2O4 141463754 EC50 = 17.13 nM T37693 C8GO7V 141463760 EC50 = 301 nM T37693 CKXG28 141463761 EC50 = 42.64 nM T37693 CZ02KM 141463762 EC50 = 969.7 nM T37693 CJY41G 141463764 EC50 = 338.2 nM T37693 C2KJ9N 141463766 EC50 = 99.86 nM T37693 C4HF2M 141463767 EC50 = 6699 nM T37693 C7AO1T 141463769 EC50 = 403.3 nM T37693 CZL4T6 141463770 EC50 = 198.8 nM T37693 C39QOI 141463775 EC50 > 10000 nM T37693 C61RIQ 141463776 EC50 = 159.4 nM T37693 C6WQI5 141463778 EC50 = 167 nM T37693 C1OY9J 141463781 EC50 = 5.701 nM T37693 C1F0BP 145949413 Ki > 10000 nM T37693 CBC13V 145949551 Ki > 10000 nM T37693 C5XM3H 145949852 Ki > 10000 nM T37693 CSI2U8 145949897 Ki > 1000 nM T37693 C1PH6E 145949978 Ki > 1000 nM T37693 CXRO20 145950071 Ki > 10000 nM T37693 CY60SW 145951064 Ki > 10000 nM T37693 CCKN03 145951123 Ki > 10000 nM T37693 CSM7J0 145951205 Ki > 10000 nM T37693 CSG0W9 145951227 Ki > 10000 nM T37693 C8EV4M 145951290 Ki > 1000 nM T37693 C4LX7H 145951404 Ki > 10000 nM T37693 C4IX1W 145951504 Ki = 7.9 nM T37693 C24POL 145951821 Ki > 1000 nM T37693 CS09YQ 145951898 Ki = 23 nM T37693 C06VUY 145951905 Ki = 606 nM T37693 C6NXD2 145952218 Ki > 1000 nM T37693 C3G5TZ 145952824 Ki > 10000 nM T37693 CS10GA 145953541 Ki > 10000 nM T37693 CDE1H5 145953638 Ki > 1000 nM T37693 CV0S3L 145953742 EC50 = 316 nM T37693 CDI42H 145953879 Ki > 10000 nM T37693 CMZ2B1 145953904 Ki = 678 nM T37693 CSHA03 145953939 IC50 = 1690 nM T37693 CZK20O 145954166 Ki = 95.5 nM T37693 C6QX5T 145954189 Ki > 10000 nM T37693 CKO9B4 145954190 Ki = 22800 nM T37693 CF63TZ 145954337 IC50 = 14670 nM T37693 COMQ03 145954409 Ki > 10000 nM T37693 C7N1JT 145954513 IC50 = 1080 nM T37693 CN7K2W 145954743 Ki > 1000 nM T37693 C03WAH 145954816 Ki > 10000 nM T37693 CVL21U 145954925 Ki = 350 nM T37693 CUE8Y2 145955444 Ki > 10000 nM T37693 C2KJ8F 145955689 Ki = 6.9 nM T37693 CX95DH 145955833 Ki > 10000 nM T37693 C46LCZ 145955918 Ki > 10000 nM T37693 CDG60N 145956233 EC50 = 280 nM T37693 CG16ZX 145956544 Ki > 10000 nM T37693 CP0L8K 145956576 Ki = 187 nM T37693 CA30EJ 145956612 Ki > 10000 nM T37693 CEX3U4 145956825 EC50 = 31 nM T37693 CX20FR 145956970 IC50 = 12620 nM T37693 C16HBG 145956992 Ki = 254 nM T37693 CX70KY 145957108 Ki > 10000 nM T37693 C1CAR4 145957287 Ki > 1000 nM T37693 CG6YU8 145957460 EC50 = 5.6 nM T37693 CR8E3C 145957540 Ki = 27.5 nM T37693 C4AUS9 145957967 EC50 = 22.5 nM T37693 CW3A0Y 145958034 Ki = 591 nM T37693 CIK3B7 145958405 Ki > 10000 nM T37693 CC5B9Y 145958428 Ki > 10000 nM T37693 C1S8TU 145958458 IC50 = 5050 nM T37693 C3IH1U 145958480 Ki > 10000 nM T37693 COP8M1 145958551 Ki > 10000 nM T37693 CEQ9W7 145958588 Ki > 10000 nM T37693 CZ1N2I 145958910 Ki > 1000 nM T37693 CATQ56 145959099 IC50 = 47710 nM T37693 C5K9TY 145959141 Ki > 10000 nM T37693 CEUL02 145959311 EC50 = 17.2 nM T37693 CDEK59 145959588 EC50 = 1.1 nM T37693 C25PYN 145959820 Ki > 1000 nM T37693 CLP94K 145960053 Ki > 1000 nM T37693 C25WFH 145960085 Ki > 10000 nM T37693 CQ3B6P 145960178 Ki > 10000 nM T37693 CVHI05 145961169 EC50 > 10000 nM T37693 CFV4A7 145962733 EC50 = 2940 nM T37693 C17TPM 145964561 Ki = 120 nM T37693 CA5S6Z 145964684 Ki > 40000 nM T37693 COB60Z 145964887 Ki > 40000 nM T37693 CHO34V 145964903 Ki = 176 nM T37693 C5L4OT 145965015 Ki = 139 nM T37693 C5RH7P 145965270 Ki > 40000 nM T37693 C47YHA 145965727 Ki > 40000 nM T37693 C09BZG 145965919 Ki > 100000 nM T37693 C5WN1R 145966442 Ki > 40000 nM T37693 C48WKZ 145966771 Ki = 12.8 nM T37693 C9ZGF6 145967019 Ki = 8.5 nM T37693 CKQU13 145967105 Ki > 40000 nM T37693 CU1O5Y 145968444 Ki > 40000 nM T37693 C0ST1H 145968723 Ki > 40000 nM T37693 C96LYC 145968771 Ki = 430 nM T37693 CNK2J9 145969213 Ki = 460 nM T37693 C0RA6B 145970762 Ki = 11.2 nM T37693 CX8I0M 145970908 Ki = 1300 nM T37693 C16RUD 145971025 Ki = 22.1 nM T37693 C5T2WE 145971274 Ki > 10000 nM T37693 C46CJZ 145971303 Ki > 40000 nM T37693 C6XAW4 145971463 Ki > 10000 nM T37693 CU3V6E 145971521 Ki = 155 nM T37693 CIU82H 145971834 Ki = 4.3 nM T37693 C92HXL 145972291 Ki > 1000 nM T37693 CDN40B 145972411 EC50 = 1.9 nM T37693 CVI92K 145972432 Ki = 329 nM T37693 CHUV20 145972574 Ki > 40000 nM T37693 CVL6X0 145972916 IC50 > 100000 nM T37693 C41SIK 145973984 Ki > 40000 nM T37693 C4G8WI 145974549 Ki > 10000 nM T37693 CR2I5X 145974580 IC50 > 10000 nM T37693 CM0ZG8 145974882 Ki > 1000 nM T37693 C09DRX 145974911 Ki > 40000 nM T37693 CEM7Z1 145975168 Ki = 6.8 nM T37693 COQP62 145975266 Ki = 2548 nM T37693 CP8A5L 145975353 Ki > 40000 nM T37693 CK8S6G 145975678 Ki > 40000 nM T37693 CFKH71 145976163 Ki = 10.4 nM T37693 C8OER4 145976515 Ki > 40000 nM T37693 C7C0GX 145976766 Ki > 1000 nM T37693 CWKV12 145976995 Ki > 40000 nM T37693 CVS75Z 145977686 Ki > 40000 nM T37693 CE9GQ8 145977936 Ki = 188 nM T37693 CKT7O8 145977995 Ki > 100000 nM T37693 C2M6BF 145978016 Ki > 1000 nM T37693 CY34IF 145978111 Ki = 52600 nM T37693 CA70FP 145978222 Ki = 286 nM T37693 CTI6J8 145978417 Ki = 24.7 nM T37693 CYAT31 145979220 Ki > 10000 nM T37693 C8PSE7 145979528 Ki = 53.9 nM T37693 C8O1FW 145979865 Ki = 581.8 nM T37693 CYAR58 145980016 Ki > 10000 nM T37693 C6P0TD 145980440 Ki > 10000 nM T37693 C4I1NP 145981357 Ki > 10000 nM T37693 CV6JC2 145981486 Ki > 10000 nM T37693 CV0Z9N 145982058 Ki > 10000 nM T37693 C65SRO 145982136 EC50 > 10000 nM T37693 C1ZD4W 145982236 Ki = 219 nM T37693 C3EAH9 145982250 Ki = 9.5 nM T37693 CGD26R 145982389 EC50 = 742 nM T37693 CXH51W 145982392 Ki > 10000 nM T37693 CLP8R3 145982513 Ki > 10000 nM T37693 CVZ8K3 145982593 Ki = 24 nM T37693 CZ8Q6U 145982659 Ki = 560 nM T37693 C9JN7H 145983146 Ki = 6.2 nM T37693 C92NMH 145983219 EC50 = 1.65 nM T37693 CP95QD 145983220 Ki = 4600 nM T37693 CGL01S 145983241 Ki = 0.4 nM T37693 C29YPO 145983245 Ki = 740 nM T37693 CP0AW6 145983324 Ki = 3000 nM T37693 CZ0O2J 145983660 EC50 = 5.4 nM T37693 CZ64LM 145983702 Ki > 10000 nM T37693 C4Y7CM 145983811 EC50 = 1.7 nM T37693 CD8SF3 145983927 Ki > 10000 nM T37693 C2O3KS 145984100 Ki = 530 nM T37693 CJ5M2I 145984210 Ki = 8.4 nM T37693 C9ILM5 145984226 EC50 = 1 nM T37693 CGO02C 145984264 Ki = 2.5 nM T37693 CI65JB 145984466 EC50 = 9.14 nM T37693 C8NI7A 145984522 Ki = 91 nM T37693 CK3PA7 145984774 Ki = 980 nM T37693 C30YIU 145984840 Ki = 1.3 nM T37693 CFL94B 145984952 Ki = 500 nM T37693 CH14SJ 145985012 Ki = 9.7 nM T37693 CWV57R 145985098 Ki = 5000 nM T37693 CF6Q7O 145985208 Ki = 6.1 nM T37693 CQ96YL 145985429 Ki = 3400 nM T37693 CUFL26 145985436 Ki = 3.7 nM T37693 C7KQ1Y 145985536 Ki = 0.7 nM T37693 CXI7F5 145985700 Ki = 5000 nM T37693 CF4P2L 145985979 Ki > 10000 nM T37693 C4T0QA 145986094 Ki = 318 nM T37693 C6N8ER 145986153 Ki = 3000 nM T37693 CC1F5K 145986420 Ki = 464 nM T37693 CW51EC 145986540 Ki > 10000 nM T37693 CQUG69 145986604 Ki > 10000 nM T37693 CS0N5V 145987144 Ki = 211 nM T37693 C96RMB 145987214 Ki > 10000 nM T37693 CHOY46 145987281 Ki = 1100 nM T37693 C6TS3J 145987421 EC50 = 18.6 nM T37693 C7EX9O 145987549 EC50 = 3400 nM T37693 CV1IH0 145988362 IC50 > 10000 nM T37693 C7K6RC 145988808 Ki > 10000 nM T37693 C5WF0E 145988921 Ki > 10000 nM T37693 C08SWB 145988974 Ki = 552 nM T37693 CDK37M 145988985 EC50 = 14.7 nM T37693 CNP5G9 145989291 Ki = 2034 nM T37693 CK74GP 145989580 Ki = 1307 nM T37693 CEK4P6 145989716 Ki > 10000 nM T37693 CD9W8O 145990481 Ki > 10000 nM T37693 C0B7HW 145990576 EC50 = 4.4 nM T37693 CK8BM3 145990869 Ki = 300 nM T37693 CL15JC 145990912 Ki = 1350 nM T37693 C0ULZ5 145990999 IC50 > 10000 nM T37693 CL7B9K 145991019 Ki > 10000 nM T37693 C4MPJ3 145991020 Ki > 10000 nM T37693 C28FLX 145991770 Ki > 10000 nM T37693 CT4GP2 145991901 Ki = 1030 nM T37693 C7R9QJ 145992065 Ki = 25 nM T37693 CZ9PB3 145993004 Ki = 200.7 nM T37693 CCH5P9 145993268 Ki = 426 nM T37693 CPBZ37 145993775 Ki = 5.7 nM T37693 CA6BY0 145993873 Ki = 990 nM T37693 CXHY67 145993892 Ki = 1969 nM T37693 CK6F7I 145994018 EC50 = 70.2 nM T37693 CYXP50 146257099 Ki = 7500 nM T37693 CR2Q4T 146257107 Ki = 3100 nM T37693 C93MHJ 146257111 Ki = 830 nM T37693 C6REF2 146257116 Ki > 10000 nM T37693 CBZ1D9 155436492 IC50 > 10000 nM T37693 CX3IL7 155436493 IC50 > 10000 nM T37693 CY2JF6 155436497 IC50 > 10000 nM T37693 CM8F5W 155436500 IC50 > 10000 nM T37693 CXIM05 155436502 IC50 > 10000 nM T37693 C3MW1Y 155436503 IC50 > 10000 nM T37693 C2NYA7 155436506 IC50 > 10000 nM T37693 CO76PL 155436509 IC50 > 10000 nM T37693 C5B8RA 155436510 IC50 > 10000 nM T37693 C2X1AI 155436512 IC50 > 10000 nM T37693 CB97LM 155436516 IC50 > 10000 nM T37693 C4NBG5 155436589 IC50 > 10000 nM T37693 CA5PI0 155436641 IC50 > 10000 nM T37693 CG3PD5 155436644 IC50 > 10000 nM T37693 CJDI76 155436645 IC50 > 10000 nM T37693 CJPO29 155436648 IC50 > 10000 nM T37693 C9WE0U 155436651 IC50 > 10000 nM T37693 CD05BE 155436652 IC50 > 10000 nM T37693 CFQ4O8 155436703 IC50 > 10000 nM T37693 CV7M3Q 155436704 IC50 > 10000 nM T37693 C2IKU4 155436706 IC50 > 10000 nM T37693 C1T7KE 155436714 IC50 > 10000 nM T37693 CG5M0C 155436719 IC50 > 10000 nM T37693 CYB9R4 155436729 IC50 > 10000 nM T37693 C3ZT6B 155436731 IC50 > 10000 nM T37693 CF9QM6 155436767 IC50 > 10000 nM T37693 C0AZ2W 155510575 Ki = 430 nM T37693 CR9G0W 155511486 EC50 > 100000 nM T37693 CJ56ZF 155511536 Ki = 212.2 nM T37693 C5BFO4 155511580 Ki = 3200 nM T37693 C4GZ8M 155512603 Ki = 20.97 nM T37693 CQ68IY 155512632 Ki = 1081.88 nM T37693 CY42GK 155512680 Ki = 12 nM T37693 CP69DA 155512716 Ki = 50.7 nM T37693 C5YR0F 155512740 Ki = 2256 nM T37693 C15NVS 155512765 EC50 = 3900 nM T37693 CBK10F 155513149 Ki = 740 nM T37693 C5LS3N 155513448 EC50 = 48 nM T37693 CG2O8Q 155513490 EC50 = 3100 nM T37693 C8W7IC 155513659 Ki = 87.1 nM T37693 C21PQJ 155514226 EC50 = 52.3 nM T37693 CXPO26 155514667 Ki > 10000 nM T37693 CC60EO 155514861 Ki = 190 nM T37693 C7HN4W 155514938 Ki > 10000 nM T37693 C5AJ0D 155515105 Ki > 7000 nM T37693 CC98DN 155515332 EC50 = 920 nM T37693 CS0C1V 155515351 Ki = 5000 nM T37693 CK2N9G 155515441 Ki = 4.28 nM T37693 CRDT78 155515622 Ki = 366 nM T37693 CV3TS9 155515668 Ki = 26 nM T37693 C5Q7TM 155515733 EC50 = 14.45 nM T37693 C8WO0D 155515901 IC50 > 10000 nM T37693 C37OWC 155516090 Ki = 20 nM T37693 CQ7KF5 155516555 Ki = 800 nM T37693 C5DPB7 155516636 Ki = 3740 nM T37693 CC0TY5 155516728 Ki = 440 nM T37693 COAX01 155516832 Ki = 1100 nM T37693 CGI38A 155516835 IC50 > 10000 nM T37693 C69WVK 155517193 Ki = 432 nM T37693 CXCY52 155517496 Ki = 1900 nM T37693 CDK74C 155517745 Ki > 10000 nM T37693 CCB70X 155518661 Ki = 150 nM T37693 CT5X0O 155519170 Ki = 6800 nM T37693 C4GY3D 155519492 Ki = 67 nM T37693 CTH10C 155519694 Ki = 92.6 nM T37693 C0HSD3 155519911 Ki = 980 nM T37693 C7N4IS 155519912 Ki > 40000 nM T37693 CCG97Q 155519954 Ki = 570 nM T37693 CKMG08 155519959 EC50 = 18.9 nM T37693 C0YW6N 155520181 Ki = 630 nM T37693 C2SV1D 155520325 Ki = 1673.74 nM T37693 CEN8W5 155520642 IC50 = 78 nM T37693 C6FQ5C 155520810 Ki > 10000 nM T37693 CCT79V 155520987 EC50 = 26400 nM T37693 COP31L 155521074 EC50 = 5400 nM T37693 CUL1B4 155521239 Ki = 1493 nM T37693 C6P2CJ 155521466 Ki = 400 nM T37693 CV0E2Y 155522138 Ki = 159.5 nM T37693 C2XB6K 155522253 EC50 = 217 nM T37693 C7NG1E 155522628 Ki > 10000 nM T37693 CV46BL 155522649 EC50 > 100000 nM T37693 C42TIR 155523370 Ki > 10000 nM T37693 C2ES7G 155523649 Ki = 70 nM T37693 CU0E6I 155523688 Ki = 4000 nM T37693 CK7RC3 155523892 EC50 = 320 nM T37693 C9VWZ8 155524523 EC50 = 3050 nM T37693 C1BUV6 155525035 EC50 = 4200 nM T37693 C0O4YW 155525197 EC50 = 189 nM T37693 CH24YB 155525250 Ki = 28700 nM T37693 CGP6I0 155525267 EC50 = 120.23 nM T37693 CAP1Q4 155525954 Ki = 2010 nM T37693 C4LEK7 155526054 EC50 > 100000 nM T37693 CP15LU 155526130 EC50 > 100000 nM T37693 CMT9X3 155526434 Ki = 38.5 nM T37693 CDY49N 155526514 Ki = 30700 nM T37693 C3NYA9 155526609 IC50 > 10000 nM T37693 C6RK9Y 155526850 Ki = 364 nM T37693 C63WYD 155527699 Ki > 10000 nM T37693 C8IEW7 155528485 Ki = 2133 nM T37693 CN8V9G 155528513 Ki > 10000 nM T37693 C5NA1U 155528573 Ki = 1010 nM T37693 C2WVB8 155529389 Ki = 2300 nM T37693 CUZ7H8 155529444 Ki > 10000 nM T37693 CRS13Y 155529582 Ki = 1.72 nM T37693 C0JOP1 155529628 Ki > 10000 nM T37693 C6T3GF 155529989 EC50 = 16100 nM T37693 C5U6KE 155530135 EC50 = 476.1 nM T37693 C7IMV5 155530567 Ki = 170 nM T37693 CT80OY 155530802 EC50 = 911 nM T37693 CS89CY 155531278 Ki = 93.3 nM T37693 C2YE4P 155531536 EC50 = 8200 nM T37693 CWLN70 155531566 EC50 > 100000 nM T37693 C6Z9GK 155531741 IC50 > 10000 nM T37693 CBG1Z4 155531768 Ki = 400 nM T37693 C9GOV6 155531899 Ki = 600 nM T37693 CPI0E3 155531980 Ki > 40000 nM T37693 CFCE85 155532563 Ki > 1000 nM T37693 CAN9V6 155533000 Ki = 4900 nM T37693 CGS63L 155533300 IC50 > 10000 nM T37693 CU5Q7F 155533412 Ki = 563.8 nM T37693 C7OKT0 155533651 Ki = 15 nM T37693 C5P4HA 155534192 EC50 = 741 nM T37693 CLG6M7 155534607 Ki > 10000 nM T37693 C5B4NZ 155535102 EC50 > 100000 nM T37693 C50YMD 155535235 Ki = 64.72 nM T37693 C1APZ8 155535329 Ki = 410 nM T37693 CA6K5I 155535568 Ki = 10000 nM T37693 CF31LR 155535617 EC50 = 58 nM T37693 CBT26P 155535766 Ki = 733 nM T37693 CMD20W 155536271 Ki = 20 nM T37693 CKI2M0 155536368 Ki = 26900 nM T37693 C3H1VC 155536420 Ki = 300 nM T37693 CDQJ85 155536760 EC50 = 4.266 nM T37693 CBK0S3 155536798 EC50 = 19 nM T37693 C7KD3W 155536933 Ki = 53.7 nM T37693 CE4L8S 155537091 EC50 = 5600 nM T37693 CBN0C9 155537341 Ki = 39.8 nM T37693 CI68ZP 155537523 Ki > 40000 nM T37693 CPT5E6 155538176 IC50 > 10000 nM T37693 CQ1PJ9 155538267 Ki = 330 nM T37693 CKM20U 155538552 Ki = 5.92 nM T37693 CA2S9E 155538637 EC50 = 5 nM T37693 CCL5E1 155538792 Ki = 97.4 nM T37693 CK2BG3 155538849 Ki > 1000 nM T37693 CWM73H 155539242 Ki > 1000 nM T37693 C3JCU0 155539433 EC50 = 5500 nM T37693 CB9MN1 155540020 Ki = 210.6 nM T37693 C7WI1O 155540156 EC50 = 707.95 nM T37693 CXRI38 155540251 Ki = 438 nM T37693 CLFP79 155540709 Ki = 845.42 nM T37693 CY5LK9 155541205 Ki = 13.5 nM T37693 C5X6EV 155541261 EC50 = 2700 nM T37693 CVRU84 155541432 Ki = 280.5 nM T37693 CYW5Z7 155542096 Ki = 280 nM T37693 CL7NT6 155542142 Ki = 26 nM T37693 C3H2LT 155542283 Ki = 110 nM T37693 C2A8JP 155542531 Ki > 10000 nM T37693 CXD78G 155543140 Ki = 120 nM T37693 CE97SK 155544312 Ki > 10000 nM T37693 CGP4Z6 155544367 IC50 = 25700 nM T37693 CB83ZR 155544851 Ki > 1000 nM T37693 C1XNB9 155545036 Ki = 133 nM T37693 C4GE0W 155545108 EC50 = 67 nM T37693 C7NA0J 155545226 Ki = 120 nM T37693 C6TDM3 155545733 Ki = 562 nM T37693 C8LD0Y 155545892 Ki = 2.7 nM T37693 C9QJF1 155546417 Ki > 10000 nM T37693 C4E5AY 155546820 Ki = 220 nM T37693 CB1RE9 155547138 Ki = 4600 nM T37693 CI51BW 155547150 Ki = 5900 nM T37693 C9GLF4 155547193 Ki = 920 nM T37693 CI1O4S 155547254 EC50 = 20200 nM T37693 CD7T4W 155547302 Ki = 272 nM T37693 C0AQU7 155547501 EC50 = 2000 nM T37693 C25LKO 155548028 Ki > 10000 nM T37693 CR4WF3 155548082 Ki = 3545 nM T37693 C9D7IV 155548445 Ki = 8.03 nM T37693 CM96DS 155548676 Ki > 1000 nM T37693 CLT98Z 155548700 Ki = 1020 nM T37693 C6TPM9 155549206 IC50 > 10000 nM T37693 C83SPR 155549297 EC50 = 104 nM T37693 CFH6B8 155549475 Ki = 210 nM T37693 CURJ67 155549486 EC50 = 116.6 nM T37693 CA8FQ3 155549571 IC50 > 10000 nM T37693 C4C0YU 155549576 EC50 = 151.36 nM T37693 CD31UY 155549880 Ki = 251 nM T37693 CM9UO8 155549886 IC50 > 10000 nM T37693 C18IUD 155550289 EC50 = 32.8 nM T37693 CPKV56 155550530 Ki = 240 nM T37693 CUZ2N8 155551511 Ki = 230 nM T37693 CC2HF0 155551585 Ki = 506 nM T37693 CDP32B 155551836 EC50 = 28100 nM T37693 CUS01D 155552044 Ki > 1000 nM T37693 CR17WN 155552557 Ki = 420 nM T37693 C0HLC1 155552734 IC50 = 36 nM T37693 CJXS06 155552844 Ki = 3000 nM T37693 CI57BL 155553206 Ki = 7.21 nM T37693 CAO59L 155553908 EC50 = 2511.8 nM T37693 CSO69Y 155554338 Ki = 525.8 nM T37693 CAG84D 155554628 Ki = 6.48 nM T37693 C5YMJ1 155554674 Ki = 3.6 nM T37693 C5D7BL 155555447 Ki = 78.7 nM T37693 CV59KM 155556037 Ki = 295.9 nM T37693 CHC64Z 155556086 IC50 > 10000 nM T37693 C6KR3O 155556171 EC50 = 14300 nM T37693 CS2G4Q 155556587 Ki > 40000 nM T37693 CU1G2L 155557132 Ki = 17400 nM T37693 CD08FU 155557245 Ki = 710 nM T37693 CH3M7N 155557426 EC50 = 5300 nM T37693 CI41HC 155557480 Ki = 9600 nM T37693 C91JPV 155557850 Ki = 2 nM T37693 CEL6Y2 155557863 EC50 = 220 nM T37693 CNJ19O 155557924 Ki > 1000 nM T37693 C5UCL8 155558472 Ki > 10000 nM T37693 C3IJF8 155558937 Ki > 1000 nM T37693 C0IOD2 155558946 Ki = 1220.19 nM T37693 C9J4CP 155559266 Ki = 208.8 nM T37693 C21FEC 155559490 Ki = 66.4 nM T37693 CRS6P3 155559856 Ki = 195.7 nM T37693 C0S4HQ 155560063 IC50 = 25.5 nM T37693 C3XL0H 155560208 IC50 > 10000 nM T37693 C20MAT 155560479 EC50 = 1200 nM T37693 CKJ7L8 155560630 Ki = 7600 nM T37693 C72BJQ 155560783 Ki = 6000 nM T37693 CY52RZ 155560863 IC50 > 10000 nM T37693 C9OJ6V 155561026 Ki = 1340 nM T37693 C27XCM 155561507 Ki = 39.6 nM T37693 C9VWA7 155561675 EC50 = 41.5 nM T37693 CS8G1A 155561709 Ki = 2070 nM T37693 C15FIN 155561744 Ki = 7300 nM T37693 C9TBR0 155562111 EC50 = 594 nM T37693 C1YK6O 155562626 EC50 = 11600 nM T37693 CX4H8P 155562737 Ki = 344 nM T37693 CU56LB 155562889 EC50 = 50 nM T37693 C84VUF 155563880 Ki = 144 nM T37693 C6GEX7 155563918 EC50 = 41900 nM T37693 C5C6ZE 155564195 Ki > 5000 nM T37693 CH7KX9 155564385 Ki = 77.3 nM T37693 CNS30G 155564805 Ki = 87.1 nM T37693 C3B9RS 155564863 Ki = 1740 nM T37693 C4F2RI 155564929 Ki > 1000 nM T37693 C2EQD9 155565124 EC50 = 48.98 nM T37693 CHC63R 155565172 EC50 = 3981 nM T37693 C18MHX 155565431 Ki = 2800 nM T37693 CG26YT 155565779 Ki = 1050 nM T37693 C7XHD5 155565941 EC50 = 4100 nM T37693 C58VGX 155565991 EC50 = 5460 nM T37693 CSC45B 155566194 Ki > 10000 nM T37693 C2NB9W 155566555 Ki = 690 nM T37693 C2Q1XD 155566691 Ki > 1000 nM T37693 CXKJ16 155566978 Ki = 1010 nM T37693 C3AWZ5 155567068 Ki = 5.3 nM T37693 CM63EC 155567324 Ki = 2500 nM T37693 C2FOQ9 155567428 Ki = 2510 nM T37693 C1SYW9 155567786 Ki > 10000 nM T37693 CR9G3I 155567842 EC50 = 520 nM T37693 CF7L0T 155568163 IC50 = 14 nM T37693 CGQT89 155568550 Ki = 59.4 nM T37693 C9R2HS 155568851 Ki = 2141.79 nM T37693 CH89DI 155569209 EC50 = 128.82 nM T37693 CP9TR0 10324985 Ki > 10000 nM T37693 C13REG 44471685 Ki = 548 nM T37693 C6MWP8 46880677 Ki = 9.6 nM T37693 C70OFQ 46880728 Ki = 35.8 nM T37693 C8NPM1 46905057 Ki = 4 nM T37693 C8AJN0 46916610 EC50 = 17.9 nM T37693 D00DNT 44452581 EC50 = 39.6 nM T37693 D00ECV 46880729 Ki = 4.5 nM T37693 D00LZJ 44452506 Ki = 154 nM T37693 D00TPO 44397641 Ki = 444 nM T37693 D00TRZ 44452580 Ki = 546 nM T37693 D00VCW 5311006 Ki = 95 nM T37693 D01IUI 44397405 Ki = 84 nM T37693 D01JHA 44431964 Ki = 17 nM T37693 D01JQX 49863581 Ki = 178 nM T37693 D01JTY 44397491 Ki = 365 nM T37693 D01JYF 325144 Ki = 1375 nM T37693 D01MCD 25059294 IC50 = 3450 nM T37693 D01MJF 44452622 Ki = 672 nM T37693 D01OFH 155160 Ki = 44 nM T37693 D01PEC 24995603 IC50 = 3400 nM T37693 D01RWS 16066912 Ki = 4270 nM T37693 D01VIA 994313 Ki = 3050 nM T37693 D01ZHW 5283389 Ki > 10000 nM T37693 D02GOH 6604822 Ki > 1000 nM T37693 D02INF 5311216 Ki = 11.8 nM T37693 D02NAW 24995605 IC50 = 12000 nM T37693 D02POA 11551123 Ki = 20 nM T37693 D02QTB 16049783 Ki = 3.3 nM T37693 D02SMK 1172084 EC50 > 30000 nM T37693 D02UEJ 44397516 Ki = 39 nM T37693 D02VSL 6918505 Ki = 0.023 nM T37693 D03DDL 44397333 Ki = 138 nM T37693 D03HFM 42617984 Ki = 190 nM T37693 D03REA 44592117 Ki = 3490 nM T37693 D03RFS 1293167 Ki > 7900 nM T37693 D03RGV 44418301 Ki = 104 nM T37693 D03SCD 44448616 Ki = 7700 nM T37693 D03SRV 44418317 Ki = 20 nM T37693 D04AMC 11559610 Ki = 1900 nM T37693 D04DQJ 72303 Ki = 5.61 nM T37693 D04ECZ 42617986 Ki = 380 nM T37693 D04EOZ 44452669 Ki = 3972 nM T37693 D04GDY 638026 Ki = 12 nM T37693 D04ICJ 1358608 Ki = 2407 nM T37693 D04LZA 44418312 Ki = 4 nM T37693 D04TSL 44452426 Ki = 1782 nM T37693 D04XGX 44592011 Ki = 2060 nM T37693 D05DFO 44406102 Ki > 10000 nM T37693 D05DXW 11616723 EC50 = 8.3 nM T37693 D05EWD 44397502 Ki = 158.85 nM T37693 D05QTX 44828492 IC50 > 10000 nM T37693 D05RGU 44406075 Ki > 10000 nM T37693 D05TQX 11702887 Ki = 8600 nM T37693 D06DTC 24995604 IC50 = 1800 nM T37693 D06EHU 11406508 Ki = 39.99 nM T37693 D06GAF 2836828 Ki < 25 nM T37693 D06JBN 5282280 EC50 = 17 nM T37693 D06JFN 1076739 Ki = 800 nM T37693 D06NXC 24996886 IC50 = 250 nM T37693 D06RIK 44406076 Ki > 10000 nM T37693 D06SKK 46918944 Ki = 553 nM T37693 D06SRX 135743701 Ki = 44.3 nM T37693 D07KZW 44418348 Ki = 29 nM T37693 D07MBC 5283454 Ki > 10000 nM T37693 D07QUV 44452688 Ki = 173 nM T37693 D08BGZ 44397406 Ki = 182 nM T37693 D08BNY 44406107 Ki = 2500 nM T37693 D08DZK 44406080 Ki > 10000 nM T37693 D08GLU 44431968 Ki = 1000 nM T37693 D08JCV 44397501 Ki = 25 nM T37693 D08JFL 44436068 Ki = 446 nM T37693 D08JYT 6483057 Ki > 1000 nM T37693 D08MON 16067266 Ki >= 10000 nM T37693 D08OAQ 44431961 Ki = 580 nM T37693 D08TXL 11584525 EC50 = 0.52 nM T37693 D08UKF 44406087 Ki > 10000 nM T37693 D08VLG 11290338 Ki = 1 nM T37693 D08YQT 2125 Ki = 110 nM T37693 D09BYO 24996885 IC50 = 4780 nM T37693 D09CKZ 9799945 Ki = 52 nM T37693 D09DSK 9799540 Ki = 0.032 nM T37693 D09FMK 4302963 Ki = 31.2 nM T37693 D09JER 44452397 Ki = 221 nM T37693 D09KFJ 44581105 EC50 = 4.6 nM T37693 D09PIQ 44418330 Ki = 23 nM T37693 D0A2BC 44452687 Ki = 421 nM T37693 D0A9PS 5281969 Ki = 160 nM T37693 D0B8AN 44418372 Ki = 169 nM T37693 D0B9RI 16067269 Ki > 10000 nM T37693 D0BS7G 5311215 Ki = 6.4 nM T37693 D0CO6T 11386747 IC50 = 4100 nM T37693 D0D4HH 44397540 Ki = 33 nM T37693 D0D6OH 104895 Ki = 0.15 nM T37693 D0D7OR 44593431 Ki = 0.9 nM T37693 D0D8PZ 93147 Ki = 63 nM T37693 D0DE9L 44418331 Ki = 9.1 nM T37693 D0DQ3F 44418313 Ki = 3.4 nM T37693 D0E0AA 24996566 IC50 > 2000 nM T37693 D0E0JU 44452623 Ki = 1120 nM T37693 D0E3ET 9950486 Ki = 0.82 nM T37693 D0E3OY 44418325 Ki = 8.2 nM T37693 D0E4OT 44452424 Ki = 700 nM T37693 D0EC6B 6443006 Ki = 52 nM T37693 D0EE0Q 44418373 Ki = 24 nM T37693 D0EX7J 49863580 Ki = 693 nM T37693 D0F3CH 11233636 Ki = 30 nM T37693 D0F3XG 44418326 Ki = 39 nM T37693 D0F4BE 11508826 Ki = 2400 nM T37693 D0F4BX 9821569 Ki = 0.15 nM T37693 D0FF6S 16038374 IC50 > 10000 nM T37693 D0FJ1I 46891225 IC50 = 2460 nM T37693 D0G2EQ 42617990 Ki = 290 nM T37693 D0G3TV 2440433 EC50 > 30000 nM T37693 D0G4VV 9893254 Ki = 0.8 nM T37693 D0G6BG 10731937 Ki >= 10000 nM T37693 D0G7GF 44431966 Ki = 44 nM T37693 D0G9EU 44452602 Ki = 3759 nM T37693 D0GD9G 44397533 Ki = 3723 nM T37693 D0GG4T 44418303 Ki = 15 nM T37693 D0I1OJ 44406101 Ki > 10000 nM T37693 D0I4AF 24992105 IC50 = 570 nM T37693 D0I4YK 6321351 Ki = 220 nM T37693 D0I7MW 44418345 Ki = 18 nM T37693 D0I9XR 11493740 EC50 = 24.4 nM T37693 D0IW4Q 44397336 Ki = 29 nM T37693 D0J3XJ 44578696 Ki = 1800 nM T37693 D0J5KA 44406095 Ki > 10000 nM T37693 D0J7CR 42617983 Ki = 150 nM T37693 D0J8KW 3081355 Ki = 0.31 nM T37693 D0K4PV 46891372 IC50 = 1280 nM T37693 D0K5DA 11502240 Ki > 10000 nM T37693 D0K7QP 44591633 Ki = 2420 nM T37693 D0K8MN 44448617 Ki = 4700 nM T37693 D0L1UA 10811495 Ki = 100 nM T37693 D0L5IM 44397559 Ki = 82 nM T37693 D0M1MQ 44397500 Ki = 7 nM T37693 D0M1ZC 44452446 Ki = 1362 nM T37693 D0N0ME 2809754 Ki = 2833 nM T37693 D0N5VO 44452649 Ki = 460 nM T37693 D0O3NY 10141893 Ki = 3.4 nM T37693 D0O4LO 23654364 Ki > 1000 nM T37693 D0O7ZJ 11461586 Ki = 6.095 nM T37693 D0O8IC 44418371 Ki = 49 nM T37693 D0OQ5H 46891330 IC50 = 801 nM T37693 D0P5VJ 10248110 Ki = 0.91 nM T37693 D0P6NA 44397671 Ki = 645 nM T37693 D0P9KU 44397635 Ki = 19 nM T37693 D0PC1Z 44452648 Ki = 639 nM T37693 D0PC5A 44243144 Ki = 7190 nM T37693 D0PE8U 25178128 Ki = 1000 nM T37693 D0Q0XV 44591632 Ki = 1630 nM T37693 D0Q4IM 44397713 Ki = 106 nM T37693 D0Q4YR 44452670 Ki = 2060 nM T37693 D0Q6FF 44397335 Ki = 20 nM T37693 D0Q8QH 11638703 Ki = 5400 nM T37693 D0Q8SO 44397464 Ki = 570 nM T37693 D0Q9FB 44418355 Ki = 33 nM T37693 D0Q9GU 1792197 EC50 > 30000 nM T37693 D0R1NR 44418349 Ki = 64 nM T37693 D0R1UA 3137700 Ki = 1.78 nM T37693 D0R3GN 44418316 Ki = 69 nM T37693 D0R6MB 46891274 IC50 = 2480 nM T37693 D0R7QF 42617989 Ki = 190 nM T37693 D0R9VY 24992763 IC50 = 5150 nM T37693 D0RI8G 44397383 Ki = 91 nM T37693 D0S2ZR 44418307 Ki = 7.1 nM T37693 D0S3UA 44418304 Ki = 6.4 nM T37693 D0T3CP 11645841 Ki = 3800 nM T37693 D0T4SE 44406097 Ki = 5100 nM T37693 D0T5WY 44418344 Ki = 41 nM T37693 D0TN1L 44418308 Ki = 62 nM T37693 D0TS5I 44418367 Ki = 25 nM T37693 D0U3ME 44300692 Ki = 2138 nM T37693 D0U4JI 44452712 Ki = 238 nM T37693 D0U5LL 2543 Ki = 16 nM T37693 D0UD9H 4302962 Ki = 4200 nM T37693 D0V0YM 24871527 IC50 = 1500 nM T37693 D0V2NQ 2385541 Ki > 7900 nM T37693 D0V3TO 44418368 Ki = 53 nM T37693 D0W9BD 44397542 Ki = 76 nM T37693 D0WD1F 44397436 Ki = 180 nM T37693 D0X0FB 44397532 Ki = 498 nM T37693 D0X1EC 44397610 Ki = 657 nM T37693 D0X1FX 49863973 Ki = 808 nM T37693 D0Y0MY 44452507 Ki = 1077 nM T37693 D0Y1MM 11710300 Ki = 81 nM T37693 D0Y6MS 44452601 Ki = 1506 nM T37693 D0Y9HT 44418338 Ki = 71 nM T37693 D0YM8O 44397465 Ki = 1353 nM T37693 D0Z1NH 42617985 Ki = 340 nM T37693 D0Z1XE 44452650 Ki = 231 nM T37693 D0Z5CX 4225440 Ki = 7900 nM T37693 D0Z6BY 44418354 Ki = 41 nM T37693 D0Z7FF 44418337 Ki = 16 nM T37693 D0Z7OB 44406064 Ki = 5200 nM T37693 D0ZL2P 16049784 Ki = 5.2 nM T37693 D0ZM1T 44250208 Ki = 10900 nM T37693 D0ZU9Z 5311257 Ki > 10000 nM T79155 CJ5E1V 119072 Ki = 37200 nM T79155 CO5Y7H 725447 Ki = 70000 nM T79155 CPJ28H 828532 IC50 = 660 nM T79155 CJ1GN3 869194 Ki = 75000 nM T79155 CBFT53 975107 IC50 = 230 nM T79155 C3X6AV 1070248 Ki = 15000 nM T79155 CQUP23 2208579 Ki = 95000 nM T79155 C97ZIP 2262135 Ki = 72000 nM T79155 C74DMH 2262990 Ki = 83000 nM T79155 CPR2F8 2931274 Ki = 50000 nM T79155 CQPJ74 2938648 IC50 = 610 nM T79155 C6WU4N 5000438 IC50 = 220 nM T79155 CV98LI 5473234 Ki = 12200 nM T79155 CI69XU 5739522 Ki = 55000 nM T79155 CDQ98U 6604561 IC50 = 20400 nM T79155 C52VYB 8072734 IC50 = 3500 nM T79155 CLG98H 25258454 Ki = 1800 nM T79155 CAF89H 25400592 IC50 = 48 nM T79155 CS9TK6 38335241 IC50 = 73000 nM T79155 CW5V7Y 44559839 IC50 = 15000 nM T79155 C0P6NY 57381616 IC50 = 68000 nM T79155 CIZ19A 57381618 Ki = 50600 nM T79155 C5L8NE 57381839 IC50 = 72000 nM T79155 C17JAZ 68284084 IC50 > 30000 nM T79155 C57MTC 70686944 Ki = 80300 nM T79155 C3I4BR 70691122 Ki = 3000 nM T79155 C15UJW 70693241 Ki = 1800 nM T79155 CQ51CP 70695325 Ki = 75100 nM T79155 C8B5HU 70695326 Ki = 77400 nM T79155 CK1OU9 76285535 Ki = 2800 nM T79155 CGO0Z1 76310236 Ki = 4400 nM T79155 CWM9B8 76310252 IC50 = 59200 nM T79155 CNA8X2 76313929 Ki = 2900 nM T79155 C2T1NM 76317472 Ki = 15600 nM T79155 C0UV9P 76317473 IC50 = 456800 nM T79155 CF8PS2 76317474 IC50 = 418300 nM T79155 COS46N 76317475 IC50 = 249300 nM T79155 CMW2Z5 76321196 Ki = 2400 nM T79155 CX3W6J 76324824 IC50 > 1000000 nM T79155 CB5G6Y 76328377 IC50 = 239000 nM T79155 C49CQJ 76328378 Ki = 2300 nM T79155 CGX1W8 76328379 Ki = 18400 nM T79155 CY25WA 76328380 Ki = 1400 nM T79155 CAEK65 76332053 IC50 = 84500 nM T79155 CZ7TH6 76335659 Ki = 15100 nM T79155 CN8O7Z 76335660 Ki = 3800 nM T79155 CKC21D 76335671 Ki = 1900 nM T79155 CY3O9X 76335672 Ki = 1300 nM T79155 CGQ90Y 118730839 IC50 = 95900 nM T79155 COLB95 118730840 IC50 = 83900 nM T79155 CGR9H8 118730843 IC50 = 80900 nM T79155 CLR3A9 118730844 Ki = 27000 nM T79155 C1UVB5 118730845 IC50 = 55700 nM T79155 C2EIU8 118730854 IC50 = 124800 nM T79155 C0SV4Z 118730863 IC50 = 135400 nM T79155 C6YQV0 118730865 IC50 = 149200 nM T79155 CKJN32 122164799 IC50 = 9000 nM T79155 C6RDX4 122192767 Ki = 16.8 nM T79155 CY0K9V 122192770 Ki = 0.8 nM T79155 CP5V4F 122225575 IC50 = 1200 nM T79155 C9USR6 134134113 IC50 = 133000 nM T79155 C34AJF 134137014 IC50 = 572000 nM T79155 C5WC3I 134143793 IC50 = 185000 nM T79155 CLW95Y 134146409 IC50 = 249000 nM T79155 CUW75P 134151146 IC50 = 272000 nM T79155 CW9NJ0 134415778 IC50 > 500 nM T79155 CCY58U 137210069 Ki = 12200 nM T79155 CPY9O5 137348758 IC50 = 820 nM T79155 CNL2Z9 137635679 Ki = 69 nM T79155 C03IMN 137647139 Ki = 130 nM T79155 CZ1H4R 137655362 Ki = 740 nM T79155 CUZ35A 138115400 IC50 > 100000 nM T79155 CE3D8P 145951877 IC50 = 22100 nM T79155 CL42TO 145953024 IC50 = 18900 nM T79155 CJZX79 145960403 IC50 = 11000 nM T79155 CCI2O5 145960428 IC50 = 940 nM T79155 CIN86F 145960836 IC50 = 6800 nM T79155 CU86EB 145960943 IC50 = 2700 nM T79155 CZO2X5 145961109 IC50 = 1900 nM T79155 CY7KI0 145961327 IC50 = 1500 nM T79155 C7X5MP 145961398 IC50 = 520 nM T79155 CZ9L2B 145961874 IC50 = 6900 nM T79155 C9GA1B 145961889 IC50 = 17000 nM T79155 CT2PO1 145961920 IC50 = 58 nM T79155 CN5HT2 145962763 IC50 = 380 nM T79155 C0UY2Z 145962805 IC50 = 11000 nM T79155 C3T4NC 145962878 IC50 = 2400 nM T79155 CX93EJ 145963112 IC50 = 2300 nM T79155 C4U7RW 145963218 IC50 = 11000 nM T79155 C1IJ2W 145963295 IC50 = 7500 nM T79155 CH7B9Y 145963477 IC50 = 5200 nM T79155 C4YH7A 145963588 IC50 = 2500 nM T79155 CXQU79 145963667 IC50 = 13000 nM T79155 C5N9AZ 145964718 IC50 > 30000 nM T79155 C7ZB3A 145965209 IC50 > 30000 nM T79155 CORX40 145965535 IC50 > 30000 nM T79155 CE18GR 145965908 IC50 = 5400 nM T79155 CD42SF 145967327 IC50 = 16000 nM T79155 CJ8Z9M 145967392 IC50 = 9000 nM T79155 C8UY7P 145967869 IC50 = 3900 nM T79155 C9VUN3 145967912 IC50 = 870 nM T79155 CB32MT 145967928 IC50 = 670 nM T79155 CL4O1U 145968107 IC50 = 940 nM T79155 C5U0VI 145968421 IC50 = 48 nM T79155 C52SCH 145968561 IC50 = 2500 nM T79155 C79ISH 145968787 IC50 = 990 nM T79155 CP9K8S 145969079 IC50 = 590 nM T79155 CD9LB5 145969087 IC50 = 450 nM T79155 CG95ZR 145969109 IC50 = 110 nM T79155 CTY2V3 145969246 IC50 = 2700 nM T79155 CK5S6B 145969453 IC50 = 4300 nM T79155 C3AJ0G 145970419 IC50 = 7000 nM T79155 C9UZ2Y 145970426 IC50 = 2800 nM T79155 C26GET 145970490 IC50 = 14000 nM T79155 CCI0T5 145970669 IC50 = 1500 nM T79155 C91KZL 145970676 IC50 = 4100 nM T79155 CK7TW6 145970889 IC50 = 5300 nM T79155 C9X3IY 145971118 IC50 = 920 nM T79155 C36ZIJ 145971366 IC50 = 30000 nM T79155 CNM9G0 145974872 IC50 = 13000 nM T79155 CYBZ02 145975368 IC50 > 30000 nM T79155 C4B8EZ 145976081 IC50 = 4500 nM T79155 C9XN7G 145976997 IC50 = 5800 nM T79155 CLR3V0 145977266 IC50 > 30000 nM T79155 CZR36C 155511554 IC50 > 100000 nM T79155 CEJC57 155512056 IC50 = 2300 nM T79155 C7JW8X 155513317 IC50 > 30000 nM T79155 CH6A8Q 155513421 IC50 = 11000 nM T79155 C3VM2R 155516045 IC50 = 9400 nM T79155 CD19EV 155517012 IC50 = 2800 nM T79155 C3M4FB 155517118 IC50 = 30000 nM T79155 C6NX4K 155519661 IC50 = 39810.72 nM T79155 C4MS1B 155519676 IC50 > 100000 nM T79155 C7S3RD 155522943 IC50 = 4700 nM T79155 CRC6L7 155524551 IC50 > 10000 nM T79155 C6L1WU 155525184 IC50 > 10000 nM T79155 CN3BH5 155527998 IC50 > 100000 nM T79155 CHYW65 155528639 IC50 > 100000 nM T79155 CD7O2G 155530095 IC50 > 100000 nM T79155 C35QWO 155531023 IC50 > 100000 nM T79155 C2X5EJ 155531124 IC50 > 10000 nM T79155 CDT7A9 155531797 IC50 > 10000 nM T79155 CBP3K1 155532687 IC50 = 4100 nM T79155 C12HON 155536142 IC50 > 100000 nM T79155 CUW43P 155537713 IC50 = 2500 nM T79155 CNB39J 155538449 IC50 = 11000 nM T79155 C8N9QK 155540725 IC50 = 1700 nM T79155 CG5J9V 155540936 IC50 = 1000 nM T79155 CY6DK3 155540964 IC50 = 39810.72 nM T79155 C29WGO 155542069 IC50 = 17000 nM T79155 CZMH45 155543862 IC50 = 10000 nM T79155 CY7DB3 155544965 IC50 = 14000 nM T79155 CX86UZ 155545827 IC50 = 2900 nM T79155 CU52QS 155545897 Ki > 10000 nM T79155 CH2S6R 155546346 Ki > 10000 nM T79155 C5MB9R 155547962 IC50 = 39810.72 nM T79155 C0JKT9 155548053 IC50 > 100000 nM T79155 CLFB25 155548371 IC50 > 100000 nM T79155 CY0AD7 155549790 IC50 = 70000 nM T79155 C93KYF 155550700 IC50 > 100000 nM T79155 COM52R 155551892 IC50 > 100000 nM T79155 CJ3FI5 155553630 IC50 > 100000 nM T79155 C3VCU1 155554104 IC50 > 30000 nM T79155 CMK57W 155554666 IC50 = 6700 nM T79155 CT9ZK6 155554786 IC50 = 14000 nM T79155 CE3G5W 155556110 IC50 > 10000 nM T79155 CJUA93 155556277 IC50 = 390 nM T79155 C0SND3 155557259 IC50 > 10000 nM T79155 CSW48V 155557718 IC50 = 79432.82 nM T79155 CTS63Q 155558248 IC50 > 10000 nM T79155 CNZ1K5 155559920 Ki > 10000 nM T79155 CZN20L 155560217 IC50 = 1900 nM T79155 C2IN3O 155560679 IC50 = 22000 nM T79155 C4CTA0 155562690 IC50 = 2500 nM T79155 CJEK04 155562801 IC50 = 24000 nM T79155 C6N0LM 155564043 IC50 > 5000 nM T79155 C32MEN 155564448 IC50 = 5700 nM T79155 CM8XB1 155565537 IC50 > 100000 nM T79155 D00LOL 970375 IC50 = 40 nM T86462 D00CSQ 5564 IC50 = 53500 nM T86462 D00HGB 4488 IC50 = 130000 nM T86462 D04AIT 5280445 IC50 = 7000 nM T86462 D05VIX 3463 IC50 = 180000 nM T86462 D06RGG 5819 IC50 = 2187.76 nM T86462 D08IFL 4037 IC50 = 50000 nM T86462 D08LFZ 3059 EC50 = 5600 nM T86462 D0B2WJ 3371 IC50 = 2900 nM T86462 D0T8VY 71771 IC50 = 170000 nM T86462 D0TG1H 3033 IC50 = 140000 nM T86462 D04DFR 11001318 IC50 = 3090.3 nM T86462 D0DK4I 4534 EC50 = 7300 nM T86462 CK1U4P 8730 IC50 = 7170 nM T86462 CBAH83 11862 IC50 = 3200 nM T86462 CC3P7O 28557 IC50 = 10000 nM T86462 CM4H7F 97032 IC50 = 1584.89 nM T86462 CJ2B1V 161924 EC50 = 6300 nM T86462 C8Y7MQ 610479 IC50 = 40000 nM T86462 CO9H7N 659923 IC50 = 1060 nM T86462 CHT4U5 677674 IC50 = 7100 nM T86462 CC36US 689075 EC50 = 67000 nM T86462 CA7H0B 693308 IC50 = 3100 nM T86462 CZ8EW9 1822412 IC50 = 20000 nM T86462 CQOR32 2816035 IC50 = 6300 nM T86462 C8YFR5 4313553 IC50 = 7700 nM T86462 CO12SM 5281790 EC50 = 21000 nM T86462 CX5J2E 5284444 EC50 = 7900 nM T86462 CAU3O8 5317238 EC50 = 23000 nM T86462 CML7U3 5353592 EC50 = 58000 nM T86462 CWQ1P8 5468215 EC50 = 11000 nM T86462 CFV8Y1 5919576 EC50 = 16000 nM T86462 C3G7DT 6365297 IC50 = 3080 nM T86462 CYP19U 9250879 IC50 = 20000 nM T86462 C9X3BW 11218587 IC50 = 11000 nM T86462 CCS9Y4 14771920 IC50 = 3070 nM T86462 CL47EC 18433807 IC50 = 1310 nM T86462 C06PCX 22133420 IC50 = 3180 nM T86462 CJM9N3 23656591 IC50 = 850 nM T86462 CBXH41 23656592 IC50 = 3160 nM T86462 CCPJ43 23656593 IC50 = 2590 nM T86462 C36LEZ 23656594 IC50 = 520 nM T86462 CZD28N 23656595 IC50 = 1360 nM T86462 CT09VW 23656596 IC50 = 475 nM T86462 C0GE9C 23656754 IC50 = 1940 nM T86462 C6W7PS 23912193 IC50 > 50000 nM T86462 C67BAF 24020163 IC50 = 6300 nM T86462 CKE3R7 44436910 IC50 = 41000 nM T86462 CF21CW 44436911 IC50 = 45000 nM T86462 C2C8YT 44436913 IC50 = 55000 nM T86462 CS6J5A 44472863 IC50 = 1960 nM T86462 C0R5ZX 44472865 IC50 = 2260 nM T86462 CV0IG8 44472866 IC50 = 2000 nM T86462 CRX2U7 44472868 IC50 = 2000 nM T86462 CV90JT 124141281 IC50 = 2020 nM T86462 CJ8G4C 134133715 IC50 = 2180 nM T86462 C0TOR6 134134052 IC50 = 1900 nM T86462 C0PB4T 134137164 IC50 = 2490 nM T86462 CEGQ24 134152257 IC50 = 2060 nM T86462 CTD7L8 134156384 IC50 = 2590 nM T86462 C9UKV8 135400370 IC50 > 50000 nM T86462 CMA49H 135406018 IC50 = 8100 nM T86462 CJ8LA2 135406035 IC50 > 50000 nM T86462 CO6M0A 135411934 IC50 > 50000 nM T86462 CD3EF5 135412515 IC50 > 50000 nM T86462 CMV5Y3 135432194 IC50 > 50000 nM T86462 CVQ6I5 135442567 IC50 > 50000 nM T86462 CKUW20 135492657 IC50 > 50000 nM T86462 CNU3X6 135541201 IC50 = 2800 nM T86462 CKC61Q 135559314 IC50 > 50000 nM T86462 C7DMH0 135755896 IC50 > 50000 nM T86462 C2AD3N 135985428 IC50 > 50000 nM T86462 CA1J2X 136180742 IC50 > 50000 nM T86462 C3F4IV 136180743 IC50 > 50000 nM T86462 C9WFH4 137287444 IC50 = 1490 nM T86462 D00RIX 5280443 IC50 = 18000 nM T86462 D05PTT 5281792 EC50 = 8600 nM T86462 D06YGF 5281787 EC50 = 8600 nM T86462 D0SP2O 7054 IC50 > 50000 nM T86462 D0U3JD 16358 IC50 = 6300 nM T86462 D0V9EN 689043 EC50 = 97000 nM T07137 D0V1UW 115355 Ki = 37 nM T07137 CB7I0S 5289053 IC50 = 85 nM T07137 C6IO2W 101913687 Ki = 10 nM T07137 C3Q4SP 101913688 Ki = 11 nM T07137 CI7L5E 118716451 Ki = 86 nM T07137 C7TN1W 118716452 Ki = 248 nM T07137 CD9E1B 118716453 Ki = 207 nM T07137 CIN42F 118716454 Ki = 79 nM T07137 CCG5N2 118716455 Ki = 74 nM T07137 C3HOL1 118716456 Ki = 173 nM T07137 C83CAL 118716457 Ki = 93 nM T07137 CK79CE 118716458 Ki = 90 nM T07137 CZI7L3 118716459 Ki = 247 nM T07137 C5FKZ1 118716460 Ki = 238 nM T07137 CGRV95 118716461 Ki = 130 nM T07137 CLH9I7 118716462 Ki = 156 nM T07137 C9OKE5 118716463 Ki = 237 nM T07137 CDB94F 118716464 Ki = 161 nM T07137 CQ1SV5 118716465 Ki = 81 nM T07137 C1E5XM 118716466 Ki = 219 nM T07137 CATC36 118716467 Ki = 87 nM T07137 C58AWJ 118716468 Ki = 177 nM T07137 C2X9QP 118716469 Ki = 109 nM T07137 C1S3NE 118716470 Ki = 19 nM T07137 CE3AS0 118716471 Ki = 15 nM T07137 C39TUB 118716571 Ki = 22 nM T07137 C8W6RV 118716572 Ki = 24 nM T07137 C0J4GN 118716573 Ki = 58 nM T07137 C2K0NW 118716574 Ki = 38 nM T07137 C8PJ9S 118716575 Ki = 20 nM T07137 C37SZQ 118716576 Ki = 14 nM T07137 CU1OV2 118716577 Ki = 13 nM T07137 CZL0E8 118716578 Ki = 34 nM T07137 C1K5AW 118716579 Ki = 31 nM T07137 CDL9H6 118716580 Ki = 34 nM T07137 C61IZC 118716581 Ki = 22 nM T07137 CXOY32 118716582 Ki = 18 nM T07137 CYBS75 118716583 Ki = 25 nM T07137 CQ65VG 118716584 Ki = 60 nM T07137 C4AUN6 118716585 Ki = 160 nM T07137 CX5KV7 118716586 Ki = 32 nM T07137 CD7Z1V 118716896 Ki = 40 nM T07137 C6RY5W 118716897 Ki = 25 nM T07137 C3AQ2F 118716898 Ki = 170 nM T07137 CA4F2U 118716899 Ki = 90 nM T07137 C3SD6V 118716900 Ki = 59 nM T07137 CVH96P 118730645 IC50 = 68 nM T07137 C9ZI2F 118730646 IC50 = 59 nM T07137 C2FNY9 118730729 IC50 = 170 nM T07137 CVUJ60 118730730 IC50 = 140 nM T07137 CN2IV3 118730731 IC50 = 130 nM T07137 C9CZK1 118730732 IC50 = 61 nM T07137 CBPD64 118730733 IC50 = 22 nM T07137 CEP7J9 118730734 IC50 = 100 nM T07137 C9X1LK 118730735 IC50 = 250 nM T07137 CZ65UC 118730736 IC50 = 130 nM T07137 CGP8J0 118730737 IC50 = 100 nM T07137 C1SZT8 118730738 IC50 = 22 nM T07137 C8FU6K 118730739 IC50 = 21 nM T07137 CG3KI4 118730740 IC50 = 64 nM T07137 CA4NK9 118730741 IC50 = 150 nM T07137 CWIZ95 118730742 IC50 = 220 nM T07137 C7PV4G 118730743 IC50 = 39 nM T07137 C6O3WB 118730744 IC50 = 40 nM T07137 CW3Q7A 118730745 IC50 = 77 nM T07137 C09ZYA 118730746 IC50 = 1030 nM T07137 CFR9K0 118730747 IC50 = 640 nM T07137 C4SOT6 118730748 IC50 = 2710 nM T07137 CE34MY 118730749 IC50 = 930 nM T07137 CZHB30 118730750 IC50 = 940 nM T07137 CJFC78 118730751 IC50 = 970 nM T07137 C5NR6K 118730752 IC50 = 990 nM T07137 CHO57A 118730753 IC50 = 990 nM T07137 CJF6H5 118730754 IC50 = 670 nM T07137 C5N2ZV 118730755 IC50 = 880 nM T07137 CF4IE5 118730756 IC50 = 940 nM T07137 C95RQA 118730757 IC50 = 970 nM T07137 CTU2R8 118730758 IC50 = 740 nM T07137 C5GT2B 118730759 IC50 = 720 nM T07137 C94EBY 118730760 IC50 = 1190 nM T07137 CS7H3I 155539271 IC50 = 422 nM T07137 CH5EM9 155541523 IC50 = 447 nM T07137 C4NYT2 155541542 IC50 = 274 nM T07137 C1DZH0 155541672 IC50 = 280 nM T07137 C2M9UW 155542673 IC50 = 266 nM T07137 C73FHE 155544224 IC50 = 63 nM T07137 C2YTZ3 155545383 IC50 = 266 nM T07137 C96POS 155547096 IC50 = 47 nM T07137 CJV42G 155547485 IC50 = 374 nM T07137 C4HQ1J 155548400 IC50 = 143 nM T07137 CV81CU 155549396 IC50 = 200 nM T07137 CCS89Y 155549408 IC50 = 147 nM T07137 CP7C5R 155549789 IC50 = 70 nM T07137 C8P4AI 155549825 IC50 = 217 nM T07137 CYK94M 155550052 IC50 = 105 nM T07137 C26BWF 155551539 IC50 = 257 nM T07137 C5ZL8G 155552614 IC50 = 335 nM T07137 CG6CT2 155553897 IC50 = 68 nM T07137 CV4T8E 155555934 IC50 = 91 nM T07137 CZFE56 155556543 IC50 = 302 nM T07137 CF13ZI 155558097 IC50 = 176 nM T07137 C16LYE 155558808 IC50 = 274 nM T07137 CM89TK 155559530 IC50 = 558 nM T07137 C61XSN 155559914 IC50 = 106 nM T07137 CU27KC 155559939 IC50 = 68 nM T07137 CO7YS3 155559958 IC50 = 168 nM T07137 C2HG7F 155559999 IC50 = 95 nM T07137 C1PXE0 155562404 IC50 = 121 nM T07137 C3E4UC 155562740 IC50 = 70 nM T07137 CE2Q1F 155563832 IC50 = 102 nM T07137 C67IDR 155565037 IC50 = 128 nM T07137 CL4QX3 155568199 IC50 = 128 nM T07137 CB5V4A 155568306 IC50 = 264 nM T48268 D0AN7B 896 EC50 = 0.069 nM T48268 D0T7OW 681 Ki = 9100 nM T48268 D0U0KW 208902 Ki = 0.045 nM T48268 D0D8FN 219018 Ki = 0.03981 nM T48268 D01ESJ 122162 Ki = 10.2 nM T48268 D0Y8UB 82148 EC50 = 0.06918 nM T48268 CHA7C3 12111 EC50 = 244000 nM T48268 CZ3LQ4 189748 Ki = 3.5 nM T48268 COT3G9 3956219 Ki = 5.3 nM T48268 CJPD17 3964826 Ki = 45708.82 nM T48268 CK8RT4 4207624 Ki = 6606.93 nM T48268 CX0OC9 5151463 Ki = 141.25 nM T48268 C8CM9B 9795837 Ki = 108 nM T48268 CXW4G5 9796251 Ki = 4.03 nM T48268 CI2A3Y 9796846 Ki = 0.153 nM T48268 C59VTY 9797460 Ki = 0.1 nM T48268 C7VG4A 9797715 Ki = 10 nM T48268 CB79WC 9798080 Ki = 0.19 nM T48268 C41QXC 9805364 Ki = 182 nM T48268 CWG0C2 9817006 IC50 = 97 nM T48268 CIL4T9 9817262 Ki = 0.13 nM T48268 C3ND5E 9817636 Ki = 0.79 nM T48268 CD3YQ2 9817692 Ki = 33 nM T48268 C89NSW 9818487 Ki = 0.37 nM T48268 CC0GV2 9819843 Ki = 1.52 nM T48268 C6K8DF 9839199 Ki = 0.068 nM T48268 CGO7V4 9839629 Ki = 0.02 nM T48268 C78CMN 9840277 Ki = 0.26 nM T48268 CDWY16 9840647 Ki = 0.17 nM T48268 C3NU4X 9850873 Ki = 13.6 nM T48268 CK8YO6 9858255 Ki = 0.06 nM T48268 C2ENY0 9859913 Ki = 4.1 nM T48268 CXO8S2 9859969 IC50 = 0.955 nM T48268 CM0LY6 9860296 Ki = 35 nM T48268 CB0R8G 9860588 Ki = 11.8 nM T48268 CO12LY 9860638 Ki = 130 nM T48268 C05WRO 9861677 IC50 = 389 nM T48268 CT5XP8 9870683 EC50 > 0.00001 nM T48268 CD9LZ7 9873402 Ki = 0.04 nM T48268 C5LQ7P 9881917 Ki = 6.8 nM T48268 C7X3QW 9883864 Ki = 0.55 nM T48268 CG1ID3 9884156 Ki = 0.69 nM T48268 C1IBZ4 9884406 Ki = 0.23 nM T48268 CT93HK 9888609 Ki = 246 nM T48268 CVR15A 9893513 Ki = 2.33 nM T48268 CO3JD2 9903515 Ki = 0.094 nM T48268 CV1CX0 9903953 Ki = 122 nM T48268 C4U7DC 9904304 Ki = 0.069 nM T48268 C8FVR1 9909783 IC50 = 9.7 nM T48268 C2O3FD 9914839 Ki = 1.74 nM T48268 C9WSM4 9916005 Ki = 0.18 nM T48268 CCUJ86 9925797 Ki = 0.39 nM T48268 CUQ86C 9925874 Ki = 26.8 nM T48268 CZJP28 9926304 Ki = 0.145 nM T48268 C6MEF3 9927219 Ki = 0.05 nM T48268 C3VE1W 9930390 Ki = 12.8 nM T48268 C0CGA4 9937825 Ki = 10.9 nM T48268 CFG16W 9947753 Ki = 0.75 nM T48268 C9SAE0 9948714 Ki = 0.55 nM T48268 C2YJC7 9970584 Ki = 1 nM T48268 C1P8AI 9998754 Ki = 0.37 nM T48268 CYT93Z 10015474 Ki = 2.3 nM T48268 CWT07A 10015475 Ki = 1 nM T48268 CM52OT 10016733 Ki = 0.19 nM T48268 CHW0S6 10016919 Ki = 0.38 nM T48268 C3W4AZ 10019103 Ki = 0.2455 nM T48268 CDZ71M 10022490 Ki = 83 nM T48268 C8JRV7 10022570 Ki = 18 nM T48268 CB8XI1 10038243 Ki = 2.2 nM T48268 C05RQN 10044270 Ki = 0.9 nM T48268 C04FNQ 10061064 Ki = 0.96 nM T48268 CT03BO 10069719 Ki = 23.7 nM T48268 CGO3N1 10089253 Ki = 16 nM T48268 CX57TO 10091075 Ki = 29 nM T48268 CKC1Y7 10163052 Ki = 6.53 nM T48268 C0IP4U 10198772 IC50 = 1000 nM T48268 CZ5I7D 10199282 Ki = 0.41 nM T48268 C7CLE4 10266979 EC50 = 2.4 nM T48268 C0HJ7G 10301190 EC50 > 0.00001 nM T48268 CZQE69 10332159 Ki = 2.8 nM T48268 C4Z6QS 10333442 Ki = 0.41 nM T48268 CGSO61 10361427 Ki = 14 nM T48268 CS5LV2 10384120 Ki = 60 nM T48268 CM8WL2 10385056 Ki = 0.11 nM T48268 C3VU0Z 10390683 Ki = 23 nM T48268 C9KLP2 10399579 Ki = 1.4 nM T48268 CJ4D8T 10400294 Ki = 2.7 nM T48268 C8HKY5 10423378 Ki = 0.44 nM T48268 C9ND1W 10424693 Ki = 1.778 nM T48268 CEZ75R 10427851 Ki = 3.4 nM T48268 C8Y7JV 10428383 Ki = 8.7 nM T48268 C5Z9GU 10446712 Ki = 0.33 nM T48268 COA8E4 10447987 Ki = 134.9 nM T48268 C1ZN2H 10452167 Ki = 0.07 nM T48268 CSUN05 10454621 Ki = 39 nM T48268 C0Y1UP 10465460 Ki = 1621.81 nM T48268 C7L8GS 10468642 Ki = 0.42 nM T48268 C32SXQ 10495702 Ki = 1.3 nM T48268 CK4P3O 10513751 Ki = 933.25 nM T48268 C6BIK5 10513752 Ki = 9332.54 nM T48268 CCM6O4 10515048 Ki = 0.093 nM T48268 CB6QE5 10517621 Ki = 17 nM T48268 C2VEM4 10518621 Ki = 17.4 nM T48268 CJ9K8Z 10518884 Ki = 7.762 nM T48268 C0YLB4 10520058 Ki = 33.9 nM T48268 CIR20T 10522674 Ki = 0.16 nM T48268 CVB47I 10522675 Ki = 0.2 nM T48268 C85RBH 10526493 Ki = 73 nM T48268 CJF51I 10540964 Ki = 0.24 nM T48268 CW1X2B 10542922 Ki = 13.2 nM T48268 CG9VZ2 10544425 Ki = 1120 nM T48268 C4B2CY 10545399 Ki = 10 nM T48268 CQ3M0U 10561982 Ki = 0.22 nM T48268 CJ6W3C 10562968 Ki = 0.12 nM T48268 CXV4U3 10563168 Ki = 645.65 nM T48268 C8FR1M 10567427 Ki = 224 nM T48268 CXW7T3 10567865 Ki = 1.66 nM T48268 CSR1Q3 10591657 Ki = 12 nM T48268 C6N2VC 10595585 Ki = 324 nM T48268 C6H7DI 10596576 Ki = 6.46 nM T48268 CC9YR3 10609620 Ki = 1445.44 nM T48268 CX6NI4 10610443 Ki = 223.87 nM T48268 C0Y8VE 10611901 Ki = 1.86 nM T48268 CQ0MA7 10616723 Ki = 0.51 nM T48268 C10KPW 10617720 Ki = 0.26 nM T48268 COE89Y 10620323 Ki = 85.1 nM T48268 COZ28S 10637638 Ki = 41.8 nM T48268 C59HRX 10638747 Ki = 354.81 nM T48268 C6M5VE 10639585 Ki = 7.586 nM T48268 C2I6TL 10640625 Ki = 17.78 nM T48268 C2L9MR 10640828 Ki = 1.59 nM T48268 CJZ06I 10641756 Ki = 5.01 nM T48268 CJK2Z3 10656443 Ki = 812.83 nM T48268 C9OI8Y 10657206 Ki = 288.4 nM T48268 CFJ95P 10658090 Ki = 102329.3 nM T48268 CQ30BW 10659603 Ki = 0.085 nM T48268 CCTW96 10661735 Ki = 0.34 nM T48268 CC0G7X 10663827 IC50 = 83 nM T48268 CZE91U 10664333 Ki = 45.7 nM T48268 C1U4EO 10666373 Ki = 117 nM T48268 C04IND 10704399 Ki = 0.51 nM T48268 CEK93Y 10704742 Ki = 4265.8 nM T48268 C38JKD 10705590 Ki = 1230.27 nM T48268 CNS05E 10709646 Ki = 36.3 nM T48268 CHE67R 10711649 Ki = 3.7 nM T48268 CB7CD3 10712600 Ki = 0.95 nM T48268 CHUL45 10712733 Ki = 0.12 nM T48268 CY3PD6 10714573 Ki = 21.9 nM T48268 CD27QT 10729569 Ki = 1.86 nM T48268 CW6XT7 10736247 Ki = 355 nM T48268 C0FN2D 10737123 Ki = 309 nM T48268 CM6K0U 10737372 Ki = 1.41 nM T48268 C27XEV 10738183 Ki = 12 nM T48268 CO2WK7 10752506 Ki = 0.22 nM T48268 CWNB23 10753255 Ki = 0.57 nM T48268 CZJL23 10754723 Ki = 1.2 nM T48268 CC7XK5 10760155 Ki = 6.31 nM T48268 C17NJY 10778397 Ki = 0.59 nM T48268 CATC31 10800029 Ki = 3.83 nM T48268 C15GYJ 10801655 Ki = 16.2 nM T48268 CP87NG 10807560 Ki = 63.1 nM T48268 CU3YN6 10808489 Ki = 5.5 nM T48268 CNM36T 10829695 Ki = 6.457 nM T48268 CRQJ04 10831675 Ki = 1.6 nM T48268 C74HBT 10850411 Ki = 0.31 nM T48268 CG74JD 10853020 Ki = 9.33 nM T48268 C2RE6J 10853021 Ki = 224 nM T48268 CT0S8G 10854190 Ki = 0.21 nM T48268 CQZ4J3 10873443 Ki = 0.77 nM T48268 C4LX0I 10882307 Ki = 0.35 nM T48268 C1O5HT 10893437 Ki = 114.82 nM T48268 CS1O3P 10903368 Ki = 275.42 nM T48268 CTS64X 10903463 Ki = 144.54 nM T48268 CQV6L3 10925379 Ki = 0.04 nM T48268 C47ROS 10925526 Ki = 2.49 nM T48268 CFZ13L 10925712 Ki = 0.02 nM T48268 C6S3NQ 10926138 Ki = 0.06 nM T48268 C7PYU9 10938056 Ki = 3.21 nM T48268 CJ52CX 10946222 Ki = 194 nM T48268 C0B4CW 10948786 Ki = 36.7 nM T48268 CXK4T2 10950593 Ki = 340 nM T48268 C6LKR7 10956792 Ki = 820 nM T48268 C7DMI9 10959837 Ki = 9.64 nM T48268 C3MU2F 10969292 Ki = 8.25 nM T48268 CAJ30W 10991315 Ki = 12.88 nM T48268 C6GJ3W 11002150 Ki = 45.71 nM T48268 CDO6V1 11002840 Ki = 0.22 nM T48268 C3YNE2 11014883 Ki = 199.53 nM T48268 C0UB2R 11045144 Ki = 245.47 nM T48268 CW7M5P 11046748 Ki = 2.76 nM T48268 C9FQH2 11058163 Ki = 141.25 nM T48268 C7EAI8 11065731 Ki = 29 nM T48268 CCW92A 11066802 Ki = 10.23 nM T48268 C0J9PL 11068422 Ki = 1.7 nM T48268 CEJZ12 11078652 Ki = 17 nM T48268 C8KO9X 11079938 Ki = 0.17 nM T48268 C6RL3D 11088627 Ki = 3.53 nM T48268 CX04WH 11098363 Ki = 10.6 nM T48268 C9R2PL 11100761 Ki = 0.047 nM T48268 CKT2U4 11109646 Ki = 79.9 nM T48268 CNS0V2 11110447 Ki = 0.21 nM T48268 CS1YX7 11131123 Ki = 18.6 nM T48268 C0CSN9 11165283 Ki = 40 nM T48268 C1Q4HG 11173131 Ki = 30.2 nM T48268 C8YVE2 11178762 IC50 = 24 nM T48268 C2C6WP 11208578 Ki = 10964.78 nM T48268 CS9ZN3 11208632 Ki = 199.53 nM T48268 CY9NP7 11213541 IC50 = 100 nM T48268 CSQB21 11219713 Ki = 89.13 nM T48268 C2U4IR 11247050 IC50 = 30 nM T48268 CK17JA 11277044 Ki = 85.11 nM T48268 CLXE76 11287002 Ki = 4570.88 nM T48268 CCND09 11304958 IC50 = 62 nM T48268 CUM40C 11304981 IC50 = 60 nM T48268 CM2EL5 11310062 Ki = 53703.18 nM T48268 C9D2WI 11314110 Ki = 6025.6 nM T48268 CQ9ZV4 11326232 Ki = 288.4 nM T48268 C8VX2J 11351216 Ki = 5.21 nM T48268 C03UAY 11361621 IC50 = 9.9 nM T48268 CT15EV 11392720 Ki = 39.81 nM T48268 C2CT0K 11393103 Ki = 38.02 nM T48268 CF20YO 11403195 Ki = 125.89 nM T48268 C31TXA 11418246 Ki = 194 nM T48268 CUE25A 11426853 Ki = 0.8913 nM T48268 CF8E2S 11430378 IC50 = 22 nM T48268 C9PW1B 11463056 Ki = 4.4 nM T48268 C12YKO 11476283 IC50 = 79 nM T48268 CDXY43 11485537 Ki = 1819.7 nM T48268 C2F8XC 11500596 Ki = 62.2 nM T48268 COR3H7 11501012 Ki = 407 nM T48268 CS9KZ5 11507534 Ki = 1.15 nM T48268 C97PGC 11515177 Ki = 33.1 nM T48268 CN4WO8 11529521 Ki = 28.9 nM T48268 CKXL24 11536746 Ki = 66.1 nM T48268 CJP73K 11536939 Ki = 0.86 nM T48268 C45FJW 11543959 Ki = 57.4 nM T48268 C90FCS 11550834 Ki = 1.02 nM T48268 C9H5ND 11573203 Ki = 138 nM T48268 C4EOD5 11581340 Ki = 2 nM T48268 CU63XE 11587169 Ki = 1.29 nM T48268 CS5A0D 11595087 Ki = 85.1 nM T48268 CIQM18 11602301 Ki = 257 nM T48268 CMQ46D 11616029 Ki = 90 nM T48268 CE75OU 11616210 Ki = 72 nM T48268 C3T9BS 11623375 Ki = 39 nM T48268 C43EBC 11624018 Ki = 3767 nM T48268 C0FTQ4 11637615 Ki = 3.3 nM T48268 C09NDO 11638009 Ki = 4.4 nM T48268 C9E1XH 11644612 Ki = 0.27 nM T48268 CNL3G5 11652196 Ki = 0.47 nM T48268 CAS86V 11666721 Ki = 58.8 nM T48268 CD48BG 11680808 Ki = 32 nM T48268 C5YRT3 11681026 Ki = 0.74 nM T48268 C9EKN8 11681201 Ki = 102 nM T48268 C1CT0E 11688043 Ki = 7.5 nM T48268 C0LR6M 11702296 Ki = 8 nM T48268 CU6A7S 11723593 Ki = 0.01 nM T48268 C0MD4I 11733059 Ki = 0.41 nM T48268 CM4UF5 11741001 Ki = 0.48 nM T48268 C25BDQ 11749479 IC50 = 5.5 nM T48268 C8LYO7 11776674 Ki = 1.738 nM T48268 CI70SF 11784134 Ki = 1.17 nM T48268 C97WON 11784859 IC50 = 120 nM T48268 CT49OP 11791741 Ki = 52.5 nM T48268 CH1YN6 11794657 Ki = 31.6 nM T48268 CDQ10E 11810280 Ki = 0.2 nM T48268 CI7SV5 11824364 Ki = 0.34 nM T48268 CRDE14 11824365 Ki = 0.5 nM T48268 CA5UO1 12004056 Ki = 19.95 nM T48268 C7X6FI 12071674 Ki = 8 nM T48268 C5TW9V 12436514 Ki = 3801.89 nM T48268 C3BJ6H 12436515 Ki = 1148.15 nM T48268 C5M9RC 12436516 Ki = 5495.41 nM T48268 C6AOC8 12985489 Ki = 1.86 nM T48268 C7IA6C 12985490 Ki = 23 nM T48268 CQS49L 12985491 Ki = 0.56 nM T48268 C24RNV 12985492 Ki = 0.71 nM T48268 C1SH0A 12985493 Ki = 0.95 nM T48268 CIP19Y 12985494 Ki = 0.52 nM T48268 CLB6Q2 12985495 Ki = 0.28 nM T48268 C8XT9Y 12985496 Ki = 48.3 nM T48268 C4DFR8 13250272 Ki = 338.84 nM T48268 CP0SV7 15453084 Ki = 0.7 nM T48268 CHEF08 15453090 Ki = 0.2 nM T48268 C5B9CQ 15453093 Ki = 2.6 nM T48268 CTC6L1 15453819 Ki = 5.9 nM T48268 CY27AW 15453821 Ki = 0.19 nM T48268 C6YB2V 16094576 Ki = 416.87 nM T48268 C46PJR 16094577 Ki = 190.55 nM T48268 C1SG9Y 16094578 Ki = 147.91 nM T48268 CHG14X 16094579 Ki = 660.69 nM T48268 C3JUF7 16094580 Ki = 6.026 nM T48268 CE46TJ 16094582 Ki = 11.48 nM T48268 CJ2F5Y 16094583 Ki = 13.18 nM T48268 C6F4KQ 16094585 Ki = 0.5248 nM T48268 C82AWU 16094586 Ki = 0.2754 nM T48268 CF3S2Z 16094587 Ki = 5.012 nM T48268 CJR8Q3 16094588 Ki = 2.63 nM T48268 CIE61K 16094591 Ki = 204.17 nM T48268 C15SJU 16094592 Ki = 524.81 nM T48268 CFLI78 16094593 Ki = 2.512 nM T48268 CY47EW 16094594 Ki = 1.549 nM T48268 C7MHQ5 16094595 Ki = 5.37 nM T48268 CFR04C 16105169 Ki = 1698.24 nM T48268 CIV2T9 16105170 Ki = 407.38 nM T48268 CU0DZ6 16656789 Ki = 0.06607 nM T48268 C0QVE3 16743123 Ki = 17.38 nM T48268 C71WVP 16743124 Ki = 70.79 nM T48268 CTP8F7 16743125 Ki = 186.21 nM T48268 CF4L3D 16743288 Ki = 407.38 nM T48268 CP30ZO 16743294 Ki = 95.5 nM T48268 C0SEN7 16743295 Ki = 11.75 nM T48268 C2BG5R 16743464 Ki = 234.42 nM T48268 CGAW53 16750566 Ki = 7.92 nM T48268 CRG52N 16750569 Ki = 0.3548 nM T48268 CI19XZ 17956989 IC50 > 10000 nM T48268 CWC8V1 17957000 IC50 = 26.3 nM T48268 CXG63C 17957007 IC50 = 4580 nM T48268 CU83BG 18007928 EC50 > 0.00001 nM T48268 C9O1UG 18007985 EC50 > 0.00001 nM T48268 CHLP82 18174996 IC50 > 10000 nM T48268 CZ2H3M 18175008 IC50 = 371 nM T48268 CE6YD4 18175028 IC50 > 10000 nM T48268 CX7D3G 18175032 IC50 = 6840 nM T48268 CAU40C 18175057 IC50 = 2000 nM T48268 C78NQP 18360631 EC50 > 0.00001 nM T48268 C0N4ZE 18360658 Ki = 16.9 nM T48268 C0DJM4 18466111 Ki = 0.034 nM T48268 C36XYE 18522208 Ki = 127 nM T48268 C2UZL1 18522267 Ki = 82 nM T48268 CE5Q1P 18522272 Ki = 95 nM T48268 C87AHP 18702059 Ki = 13 nM T48268 CRO46J 19703015 Ki = 1.2 nM T48268 C1I0OZ 19703063 Ki = 117 nM T48268 CS2VZ6 20355585 Ki = 2.2 nM T48268 CS5KB7 20590652 Ki = 2 nM T48268 C8KEI5 20590653 Ki = 5 nM T48268 CDXF27 20590654 Ki = 2 nM T48268 C6V1TU 20590664 Ki = 90 nM T48268 CNS15E 20590665 Ki = 90 nM T48268 CEM7F6 20642483 Ki = 2.8 nM T48268 CL64ZO 21581653 Ki = 35 nM T48268 C90HJK 21581654 Ki = 0.3 nM T48268 C6ZQD8 21916760 IC50 = 879 nM T48268 CZ2AW7 22004791 Ki = 0.022 nM T48268 CD6V5I 22004862 Ki = 0.0065 nM T48268 C1AX5C 22037991 IC50 = 44 nM T48268 CO4A0H 22375366 IC50 = 3 nM T48268 CO1L6H 22375370 IC50 = 2.3 nM T48268 CVJX25 22375372 IC50 = 1.5 nM T48268 CU4T2X 22375392 IC50 = 3.1 nM T48268 C90OUD 22375402 IC50 = 75 nM T48268 CIE2B1 22375407 IC50 = 94 nM T48268 C6CQ5D 22375417 IC50 = 32 nM T48268 CELS26 22718521 Ki = 35 nM T48268 CS3WC4 22718530 Ki = 89 nM T48268 C5FD7I 22718548 Ki = 57 nM T48268 CS4IY9 22718555 Ki = 88 nM T48268 C7FX6M 22718571 Ki = 22 nM T48268 CZ6D9B 22718576 Ki = 5.3 nM T48268 CRQT08 22718579 Ki = 35 nM T48268 CR46PF 22718585 Ki = 15 nM T48268 C4XJ6L 22718596 Ki = 17 nM T48268 CM6ZG9 22718602 Ki = 4.5 nM T48268 CEC0I5 22718610 Ki = 10 nM T48268 CB2QJ0 22718619 Ki = 16 nM T48268 CR5D8T 22718654 Ki = 29 nM T48268 CSPB82 22718661 Ki = 27 nM T48268 CL4CF8 23642306 EC50 = 2.754 nM T48268 C9U6TM 23642307 Ki = 0.537 nM T48268 CG78OH 23658143 EC50 = 25.12 nM T48268 CY68EQ 23658144 EC50 = 0.7943 nM T48268 CBS59I 23658145 Ki = 5.495 nM T48268 CLJ03E 23658146 Ki = 0.3162 nM T48268 C3X5PA 24750069 Ki = 0.7586 nM T48268 CPLG20 24750070 Ki = 7.413 nM T48268 C6NQP2 24750071 Ki = 0.1047 nM T48268 CUZ3C2 24750077 Ki = 0.02754 nM T48268 C67HYD 24750188 Ki = 0.871 nM T48268 C51VEA 24750189 Ki = 0.1122 nM T48268 CAV48F 24750190 Ki = 3.89 nM T48268 CQD54L 24750191 Ki = 0.1995 nM T48268 CYQ6A7 24750193 Ki = 1.995 nM T48268 CYFL67 24750194 Ki = 3.715 nM T48268 CO87FN 24750195 Ki = 52.48 nM T48268 CK0AC4 24954990 Ki = 0.22 nM T48268 C8A5QN 24954991 Ki = 0.53 nM T48268 CZE7M2 24954992 Ki = 0.93 nM T48268 CRU4L6 24955342 Ki = 6.1 nM T48268 CQFI43 24955343 Ki = 0.085 nM T48268 CFPI79 25014882 IC50 = 5900 nM T48268 C21GCY 25022429 Ki = 7.8 nM T48268 C8K5GJ 25022442 Ki = 60.26 nM T48268 C6P0QW 25209860 Ki = 14 nM T48268 C8E9JX 25209861 Ki = 8 nM T48268 CLW71G 25209998 Ki = 7.079 nM T48268 CGSV97 25209999 Ki = 30 nM T48268 C4RPN9 25210000 Ki = 26.3 nM T48268 C7WY8N 25210131 Ki = 14.45 nM T48268 CFU8K9 25210132 Ki = 0.001 nM T48268 C96ZPF 25210133 Ki = 14.79 nM T48268 C54OEZ 25210134 Ki = 24.55 nM T48268 CJQX17 25210135 Ki = 117.49 nM T48268 CM93GU 25270146 Ki = 2.6 nM T48268 CY1K7H 44241665 Ki = 6.918 nM T48268 CRE65K 44241666 Ki = 2.291 nM T48268 CFB6X3 44264689 Ki = 64 nM T48268 CG8OF4 44264692 Ki = 84 nM T48268 C15DKZ 44264705 Ki = 0.39 nM T48268 CN0ZJ8 44264706 Ki = 1.8 nM T48268 C6Z7EG 44264707 Ki = 4.2 nM T48268 CUOG79 44264769 Ki = 0.1 nM T48268 CUSJ15 44264818 Ki = 0.12 nM T48268 C8K7XE 44264843 Ki = 7.2 nM T48268 CJNR68 44264844 Ki = 4.8 nM T48268 CI0PL7 44264849 Ki = 5.5 nM T48268 C6XF9C 44264857 Ki = 250 nM T48268 C1GKR5 44264861 Ki = 0.49 nM T48268 C5GKS4 44264871 Ki = 0.68 nM T48268 CJIZ29 44264892 Ki = 0.17 nM T48268 CCXI31 44264903 Ki = 0.23 nM T48268 CKV1H3 44264904 Ki = 0.71 nM T48268 CLQ9O0 44264909 Ki = 0.78 nM T48268 C5U1EH 44264942 Ki = 4.7 nM T48268 CJUS17 44264949 Ki = 0.75 nM T48268 C3HKR4 44264950 Ki = 15 nM T48268 CF82IP 44264962 Ki = 2.1 nM T48268 CNXG58 44264964 Ki = 110 nM T48268 C32BSH 44264965 Ki = 150 nM T48268 CP9SA3 44264982 Ki > 400 nM T48268 CF59MU 44264983 Ki = 39 nM T48268 CHQ94P 44272252 IC50 = 103 nM T48268 CMN1U0 44272305 Ki = 1.9 nM T48268 C0LX2R 44272316 Ki = 0.24 nM T48268 C93HVQ 44272317 Ki = 0.14 nM T48268 C0VD1G 44272320 Ki = 0.08 nM T48268 CQ01LK 44272334 Ki = 0.28 nM T48268 C6NR1W 44272335 Ki = 0.04 nM T48268 CZBX31 44272406 Ki = 2.2 nM T48268 C6LP4B 44272410 Ki = 0.13 nM T48268 C60OAS 44272422 Ki = 0.75 nM T48268 C2BW8J 44272424 Ki = 12.6 nM T48268 CUX94M 44272425 Ki = 2.2 nM T48268 CUJ30W 44272430 Ki = 0.32 nM T48268 C5SVO1 44272431 Ki = 1.2 nM T48268 CO1GB4 44272438 Ki = 2.5 nM T48268 CQ9L6O 44272440 Ki = 0.88 nM T48268 CP1OX9 44272443 Ki = 0.8 nM T48268 C0L7ME 44272444 Ki = 1 nM T48268 C1B9MP 44272451 IC50 = 224 nM T48268 C4SXT1 44272486 IC50 = 1.5 nM T48268 CCW2B6 44272487 IC50 > 1000 nM T48268 C8GYN2 44272497 IC50 > 1000 nM T48268 CZU41O 44272520 IC50 > 1000 nM T48268 CLPA83 44272521 IC50 = 90 nM T48268 C69SPD 44272539 IC50 = 270 nM T48268 CO76HL 44272589 IC50 > 1000 nM T48268 C8MZP1 44272590 IC50 > 1000 nM T48268 CB82FD 44272591 IC50 = 1.6 nM T48268 CI3WK7 44309030 Ki > 1000 nM T48268 C67MUK 44309034 Ki > 1000 nM T48268 C2ID4J 44317725 Ki = 6.7 nM T48268 CQ7C3V 44317822 Ki = 16 nM T48268 CF8K5Q 44317845 Ki = 1.2 nM T48268 C3TBX1 44348996 Ki = 4.7 nM T48268 CMF80O 44349100 Ki = 22 nM T48268 CV9M5R 44349171 Ki = 12 nM T48268 CW9I4V 44349258 Ki = 26 nM T48268 C3OJ1M 44349269 Ki = 52 nM T48268 CDJ7X9 44349270 Ki = 114 nM T48268 C5DGU1 44349294 Ki = 61 nM T48268 CSA4U3 44349305 Ki = 38 nM T48268 CC92NR 44349329 Ki = 36 nM T48268 CW6U7K 44349362 Ki = 7.6 nM T48268 CLTG60 44353165 Ki = 0.18 nM T48268 CUQE30 44357899 Ki = 22.3 nM T48268 CYT31X 44358035 Ki = 39.3 nM T48268 CEB6M2 44358087 Ki = 85 nM T48268 CWT62A 44358088 Ki = 121 nM T48268 C9SHE8 44358146 Ki = 0.31 nM T48268 CPE31J 44358184 Ki = 1 nM T48268 CR21BK 44358196 Ki = 0.4 nM T48268 C4RVX3 44358217 Ki = 19 nM T48268 CTXM75 44358218 Ki = 5.8 nM T48268 CQE7S2 44358231 Ki = 2.1 nM T48268 C9JGW6 44358238 Ki = 4.6 nM T48268 CGR39W 44358274 Ki = 0.94 nM T48268 CTE2X3 44358275 Ki = 10.8 nM T48268 CSY8C4 44358276 Ki = 2.6 nM T48268 C3AJU1 44358312 Ki = 6.4 nM T48268 CK12OG 44359437 Ki = 13.8 nM T48268 C2O1DS 44389768 Ki = 90 nM T48268 CHS49R 44389812 Ki = 20 nM T48268 C5RTM7 44389813 Ki = 30 nM T48268 C4TYV6 44389839 Ki = 40 nM T48268 C0CD8U 44389845 Ki = 30 nM T48268 C6ZMD5 44389864 Ki = 40 nM T48268 C2LOD6 44394338 Ki = 98 nM T48268 CKY2H1 44394394 Ki = 33 nM T48268 C64MHD 44394415 Ki = 10 nM T48268 C40JFL 44394416 Ki = 54 nM T48268 CW4I0M 44394435 Ki = 10 nM T48268 C2ZOS9 44394438 Ki = 2.8 nM T48268 C06JWG 44394456 Ki = 52 nM T48268 CRDH82 44394478 Ki = 162 nM T48268 CDN4K0 44394508 Ki = 7.2 nM T48268 CO61EF 44394532 Ki = 14 nM T48268 CY4CN6 44394535 Ki = 6 nM T48268 C2SKD1 44394556 Ki = 152 nM T48268 CD0XI1 44395856 IC50 > 1000 nM T48268 CRS38H 44395895 IC50 > 1000 nM T48268 C8V2YE 44395896 IC50 = 140 nM T48268 C6CO1Q 44395915 IC50 = 45 nM T48268 C83XAQ 44395939 IC50 = 280 nM T48268 C5U4JB 44395994 IC50 = 370 nM T48268 C0WEC1 44396034 IC50 = 240 nM T48268 C8JB0P 44396057 IC50 = 24 nM T48268 CBMP19 44396058 IC50 = 220 nM T48268 C4L1DA 44396073 IC50 = 400 nM T48268 CE52QV 44396074 IC50 = 76 nM T48268 C4JX9C 44396100 IC50 = 810 nM T48268 C1JXG0 44396113 IC50 = 1000 nM T48268 CT8LC6 44396135 IC50 > 1000 nM T48268 CZF6N7 44396136 IC50 = 270 nM T48268 CI2WG8 44396148 IC50 = 160 nM T48268 CNT8E5 44396149 IC50 = 130 nM T48268 CA9ZH4 44412063 Ki = 1445 nM T48268 C7Y1FX 44412078 Ki = 1259 nM T48268 CN65SG 44412079 Ki = 1047 nM T48268 C9ZLR7 44412082 Ki = 1738 nM T48268 CMD54S 44412141 Ki = 2344 nM T48268 CN9Y8X 44424017 Ki = 14.3 nM T48268 CPU57Y 44424018 Ki = 62.4 nM T48268 C2L0YH 44424019 Ki = 65.02 nM T48268 C1S7IT 44424020 Ki = 7.75 nM T48268 CJ80GI 44424021 Ki = 15.43 nM T48268 CT4C0R 44424022 Ki = 44.01 nM T48268 CHOU45 44424023 Ki = 4.8 nM T48268 C0EZV4 44424024 Ki = 20 nM T48268 C18YWB 44424025 Ki = 7290 nM T48268 C5NFQ7 44424026 Ki = 573 nM T48268 CXT3N5 44426096 Ki = 1.4 nM T48268 C0YUF3 44429441 Ki = 1.738 nM T48268 C8UYO4 44429442 Ki = 1.096 nM T48268 C7DGK2 44429443 Ki = 0.6761 nM T48268 CXP8Z1 44429444 Ki = 1.549 nM T48268 CH79WZ 44429445 Ki = 2.63 nM T48268 CW7B9P 44429446 Ki = 1.349 nM T48268 CY7WU6 44429447 Ki = 0.6761 nM T48268 CNDQ75 44429448 Ki = 0.537 nM T48268 CE1X8B 44429449 Ki = 1.318 nM T48268 CU2Y3J 44429450 Ki = 2.291 nM T48268 CG42LM 44429451 Ki = 2.138 nM T48268 C39FXQ 44429452 Ki = 3019.95 nM T48268 C6P4GD 44429453 Ki = 616.6 nM T48268 CQ9VS6 44429454 Ki = 870.96 nM T48268 CRY10T 44429455 Ki = 457.09 nM T48268 C63DEA 44429456 Ki = 676.08 nM T48268 CE49OW 44429457 Ki = 851.14 nM T48268 CQ37OL 44436051 Ki = 12.59 nM T48268 C69IKT 44576399 IC50 > 1000 nM T48268 CCP3T7 44576404 IC50 > 10000 nM T48268 CIQX03 44576405 IC50 > 10000 nM T48268 C74LMW 44576406 IC50 = 5320 nM T48268 C0LV5I 44579115 EC50 = 0.5 nM T48268 C5VU7G 44579163 Ki = 0.94 nM T48268 C8R3KQ 44579164 Ki = 8.3 nM T48268 C1Y3GP 44579259 Ki = 0.42 nM T48268 C2R4MV 44579260 Ki = 0.64 nM T48268 CPAD41 44579261 Ki = 43.3 nM T48268 CBYC81 44579296 Ki = 7.54 nM T48268 C40IDJ 44581851 Ki = 0.11 nM T48268 C8NO1P 44587356 Ki = 33.6 nM T48268 CB2ZQ5 44587357 Ki = 36.2 nM T48268 CR59BF 44593609 IC50 > 10000 nM T48268 C8S0ZG 44593610 IC50 = 560 nM T48268 CD4G5Y 45267465 Ki = 660.69 nM T48268 CV7Y5J 45268303 Ki = 7.762 nM T48268 C7LNE2 45268309 Ki = 223.87 nM T48268 CV5KC1 45268310 Ki = 63 nM T48268 CS04YH 45268318 Ki = 891.25 nM T48268 CDW89L 45269177 Ki = 85.11 nM T48268 CNC8W0 45269183 Ki = 42.66 nM T48268 C3UAM7 45270052 Ki = 9 nM T48268 C09LCX 46845151 Ki = 59.1 nM T48268 C3ID6J 46865422 EC50 = 0.05 nM T48268 C9Y6JN 46884550 Ki = 102 nM T48268 CE3S8R 46884551 Ki = 0.0326 nM T48268 CV97RU 46884552 Ki = 1.61 nM T48268 CZ1AK8 46884553 Ki = 0.00069 nM T48268 C2L9TZ 46884554 Ki = 69.3 nM T48268 CY6X5U 46884555 Ki = 121 nM T48268 C98CGH 46884599 Ki = 105 nM T48268 CQAF97 46885226 Ki = 0.04705 nM T48268 CI7Q8L 46885227 Ki = 0.00055 nM T48268 CUF3Q1 46885228 Ki = 0.00103 nM T48268 CA6V4P 46885229 Ki = 2300 nM T48268 CP06TV 46885286 Ki = 13.4 nM T48268 CU92VL 46885287 Ki = 72.2 nM T48268 CY0JL9 46885288 Ki = 27.9 nM T48268 COK9Z0 46888491 EC50 > 0.00001 nM T48268 C1XUG9 46888492 EC50 > 0.00001 nM T48268 C2EJD1 46888520 EC50 > 0.00001 nM T48268 CLKO39 46888521 EC50 > 0.00001 nM T48268 CQ51ZE 46888522 Ki = 4.22 nM T48268 C29LQB 46919520 EC50 = 1697 nM T48268 C4X2NV 46935149 Ki = 263.03 nM T48268 C1ZYJ3 46935150 Ki = 4.365 nM T48268 CW2KQ0 49862664 EC50 = 2100 nM T48268 C1X3WL 49862665 EC50 = 342.9 nM T48268 CG78ZY 49862736 EC50 = 115 nM T48268 C8GVY6 49862737 EC50 = 735 nM T48268 C0N8IJ 49862738 EC50 = 295 nM T48268 C5MZ9X 49862739 EC50 = 465 nM T48268 CBIK17 49862740 EC50 = 615 nM T48268 C13BFO 49865147 Ki = 12589.25 nM T48268 CG5X2S 49865148 Ki = 5128.61 nM T48268 CABU10 49865149 Ki = 9.55 nM T48268 C8F7NS 49865203 Ki = 109.65 nM T48268 CQW04N 49865204 Ki = 4.677 nM T48268 C71VAK 49865205 Ki = 660.69 nM T48268 CAYG40 49865206 Ki = 7.079 nM T48268 C91NRX 49865265 Ki = 39.81 nM T48268 C5ZKD6 49865266 Ki = 2398.83 nM T48268 C8AHB3 49865267 Ki = 501.19 nM T48268 C9NR2L 49865268 Ki = 12.88 nM T48268 C2SM4J 49865269 Ki = 20.89 nM T48268 C8LI9V 49865270 Ki = 9.772 nM T48268 C96QKF 49865317 Ki = 48.98 nM T48268 CH9AZ5 49865318 Ki = 6.761 nM T48268 CQ08DG 49865319 Ki = 3.715 nM T48268 CNJ1M3 49865320 Ki = 67.61 nM T48268 CK6MU2 49865321 Ki = 2.754 nM T48268 C5PYK1 49865322 Ki = 5.012 nM T48268 CL4WG7 49865323 Ki = 26.3 nM T48268 CJRE71 49865324 Ki = 6.026 nM T48268 C8HN7M 49865373 Ki = 346.74 nM T48268 CTYD96 49865374 Ki = 4897.79 nM T48268 C10JEM 49865375 Ki = 302 nM T48268 CQ1X4S 49865376 Ki = 1318.26 nM T48268 CIET97 49865377 Ki = 12302.69 nM T48268 CA2B5F 49865378 Ki = 263.03 nM T48268 CR2E8T 49865423 Ki = 6760.83 nM T48268 C4EO5K 49865424 Ki = 64565.42 nM T48268 CDX4B0 49865425 Ki = 4365.16 nM T48268 C9LX2O 52918077 Ki = 0.6 nM T48268 CP7A1S 52918078 Ki = 0.28 nM T48268 C87COQ 52918079 Ki = 0.3 nM T48268 CJ7IF1 52918080 Ki = 0.68 nM T48268 C8NWT6 52953165 Ki = 0.24 nM T48268 CY5R6B 53231366 EC50 = 0.64 nM T48268 CLNE80 53231367 Ki = 24.8 nM T48268 CU79SK 53231464 Ki = 10.7 nM T48268 C7ZJH2 53231465 EC50 = 0.68 nM T48268 CW9OF1 53237946 Ki = 0.018 nM T48268 C58MYW 53237947 Ki = 0.011 nM T48268 CO3XJ2 53237948 Ki = 0.035 nM T48268 C7AF5C 53237949 Ki = 0.01 nM T48268 CP18VR 53237950 Ki = 0.084 nM T48268 CR9LF5 53237951 Ki = 0.0085 nM T48268 CW9G3R 53238182 Ki = 0.0067 nM T48268 C7N6RW 53238183 Ki = 0.014 nM T48268 CU27MO 53238184 Ki = 0.0096 nM T48268 CF1OY4 53238185 Ki = 0.034 nM T48268 CB3H8J 53238186 Ki = 0.02 nM T48268 C3AG1Y 53238407 Ki = 0.009 nM T48268 CB12VT 53238408 Ki = 0.037 nM T48268 C2S0AN 53238409 Ki = 0.34 nM T48268 C67VCY 53238410 Ki = 0.011 nM T48268 C0B2SG 53238411 Ki = 0.77 nM T48268 C12UVM 53238412 Ki = 0.006 nM T48268 C5KW2F 53310838 Ki = 4.5 nM T48268 C92HTZ 53310839 Ki = 0.19 nM T48268 CCA16D 53310840 Ki = 0.28 nM T48268 C53MGN 53310841 Ki = 0.14 nM T48268 CM9A6H 53310987 Ki = 0.33 nM T48268 CT7HJ5 53827707 IC50 = 6.7 nM T48268 C5Q4SP 54581170 Ki = 5 nM T48268 CC8U1V 54582194 Ki = 742 nM T48268 C0W8TR 54582195 EC50 = 10 nM T48268 CMD87P 54583161 Ki = 7440 nM T48268 C3ANK6 54583162 Ki = 1090 nM T48268 CMP96I 54584154 Ki > 10000 nM T48268 C6G3KX 54584155 Ki = 4007 nM T48268 C0X1MI 54586060 Ki = 550 nM T48268 C6MWF0 54586061 Ki = 929 nM T48268 CO03ZV 54770909 Ki = 7980 nM T48268 C7KP3U 56653119 Ki = 0.19 nM T48268 C2RLP3 56653120 Ki = 49 nM T48268 CYL23N 56653479 Ki = 87 nM T48268 C2AVC9 56659223 Ki = 0.2 nM T48268 CH1IR9 56661499 Ki = 2089.3 nM T48268 CV2RN0 56661512 Ki = 1000 nM T48268 CG7H2A 56662798 Ki = 309.03 nM T48268 C5WP1S 56662799 Ki = 245.47 nM T48268 CCQ27N 56664925 Ki = 181.97 nM T48268 CXGW49 56671856 Ki = 93.33 nM T48268 C6OCQ1 56671857 Ki = 158.49 nM T48268 CZ56WJ 56671858 Ki = 36.31 nM T48268 C17XRI 56678563 Ki = 812.83 nM T48268 CJU8R5 56681902 Ki = 40.74 nM T48268 CDW2N1 71508232 Ki = 0.073 nM T48268 CGS73W 71508233 EC50 = 0.024 nM T48268 CWO72Z 71508235 EC50 = 0.2 nM T48268 CP3Q5Z 71533430 Ki = 0.03 nM T48268 C6ZE5N 71540275 Ki = 6.8 nM T48268 C92WJY 71540389 Ki = 0.09 nM T48268 C0NZ2T 71540390 Ki = 86 nM T48268 CM76EA 76313971 Ki = 10 nM T48268 CMD3V9 76317510 Ki = 26 nM T48268 CR75IF 76317511 Ki = 315 nM T48268 CS1ZW2 76332093 Ki = 96 nM T48268 CF23TN 79374977 Ki > 10000 nM T48268 C6KAF4 81689735 Ki = 190 nM T48268 C3M7TG 85880795 Ki = 21.4 nM T48268 CG0V6I 86272984 Ki = 220 nM T48268 C3GYF8 86272986 Ki = 560 nM T48268 C82OPI 86272988 Ki = 535 nM T48268 CHK4C2 86272990 Ki = 160 nM T48268 CU78IJ 86273221 Ki > 1000 nM T48268 C2EK6O 86273222 Ki = 44 nM T48268 CBL0V9 86273223 Ki > 1000 nM T48268 CSC62G 86273226 Ki = 1 nM T48268 CDG2J4 86273227 Ki = 3.8 nM T48268 CY4N2D 86273228 Ki = 0.45 nM T48268 CJHY29 86273229 Ki = 4.9 nM T48268 CT6U5G 86273470 Ki = 498 nM T48268 CHMV24 90655902 Ki = 0.29 nM T48268 CAT42J 90666302 Ki = 21.38 nM T48268 CBF12L 90666303 Ki = 5.754 nM T48268 CHY40Z 90666304 Ki = 81.28 nM T48268 CFMG86 90666305 Ki = 2.239 nM T48268 C1W2ZM 90666306 Ki = 3.715 nM T48268 CB4TU6 90666307 Ki = 9.333 nM T48268 CM98LH 90666308 Ki = 33.88 nM T48268 CVR1U5 90666309 Ki = 199.53 nM T48268 C4FMX7 102361822 EC50 = 383000 nM T48268 CJR85X 118712349 Ki > 10000 nM T48268 CKM9T6 118712350 Ki > 10000 nM T48268 CCY6M7 118712351 Ki > 10000 nM T48268 CM40LO 118712352 Ki > 10000 nM T48268 CFK26G 118712353 Ki > 10000 nM T48268 C4QAV9 118712354 Ki > 10000 nM T48268 C5TK7E 118712355 Ki > 10000 nM T48268 C42HKY 118712356 Ki > 10000 nM T48268 CB2RV5 118712357 Ki > 10000 nM T48268 C9Q5MI 118712358 Ki > 10000 nM T48268 C7C6SW 118712359 Ki > 10000 nM T48268 CVA4W3 118712360 Ki = 380 nM T48268 CZ7HD5 118712361 Ki > 10000 nM T48268 C1INH7 118712362 Ki > 10000 nM T48268 CWV7N2 118712363 Ki > 10000 nM T48268 C8V6WQ 118712364 Ki > 10000 nM T48268 CH9BF2 118712365 Ki > 10000 nM T48268 CKG94Y 118712366 Ki > 10000 nM T48268 CR51PL 118712367 Ki > 10000 nM T48268 CTQ8O1 118712368 Ki > 10000 nM T48268 C2G3AN 118712369 Ki > 10000 nM T48268 CGF6R8 118712370 Ki > 10000 nM T48268 CKF3O6 118712371 Ki > 10000 nM T48268 C0X1MH 118712372 Ki = 190 nM T48268 C9AOZ2 122178507 Ki = 16 nM T48268 C7YDM4 122178508 Ki = 68 nM T48268 CZMA87 122178509 Ki = 4 nM T48268 C60SIG 122178510 Ki = 530 nM T48268 CNI19Q 122178511 Ki > 1000 nM T48268 C1NI7Q 122178512 Ki > 1000 nM T48268 C73KSA 122178513 Ki = 17 nM T48268 CPT16O 122193492 Ki = 3.4 nM T48268 CV5L0S 122220128 Ki = 0.3467 nM T48268 CWV9T8 127025170 Ki = 46 nM T48268 CU67PG 127025781 EC50 = 5.8 nM T48268 C0SAG6 127025782 EC50 = 8.8 nM T48268 CG53JK 127025783 Ki = 2.1 nM T48268 C7P8JY 127025784 Ki = 0.7 nM T48268 CK92ZA 127025786 EC50 = 6.2 nM T48268 C3YG1L 127025787 Ki = 4.2 nM T48268 C56JXR 127025788 Ki = 0.8 nM T48268 CL24NY 127026062 Ki = 0.4 nM T48268 CC87HM 127026423 Ki = 0.09 nM T48268 C7Z0HG 127026424 Ki = 1.7 nM T48268 CBHW31 127026425 EC50 = 8.8 nM T48268 C4CFA1 127026426 EC50 = 3.2 nM T48268 CQ85ZK 127026427 Ki = 0.6 nM T48268 C3EA0C 127027022 Ki = 7 nM T48268 CB8RL9 127029516 Ki = 0.7 nM T48268 C4C7RU 127038129 Ki = 1.778 nM T48268 CY2JR9 127038130 Ki = 9 nM T48268 CU1KI9 127038131 Ki = 43.65 nM T48268 CO45XY 127038132 Ki = 8.913 nM T48268 CV0C2N 127038225 Ki = 9 nM T48268 CDV69R 127039212 Ki = 1.3 nM T48268 C2HQC8 127039218 Ki = 59 nM T48268 CYKA08 127040021 Ki = 0.09 nM T48268 C90XDV 127040022 Ki = 5 nM T48268 CPC79R 127040355 Ki = 5 nM T48268 C9RW7G 127041168 Ki = 7.762 nM T48268 CLK51B 127041169 Ki = 8.1 nM T48268 CYKA14 127041170 Ki = 14.45 nM T48268 CW73LQ 127042142 Ki = 0.14 nM T48268 CS0H8W 127042442 Ki = 0.03 nM T48268 COC3L8 127042791 Ki = 0.08 nM T48268 CFS87E 130400672 Ki = 110 nM T48268 CF1EZ3 137631636 Ki = 0.48 nM T48268 CR21JG 137633839 Ki = 73 nM T48268 CW39EH 137636079 Ki = 1 nM T48268 C6F1NM 137636173 Ki = 0.3 nM T48268 C7RUG3 137636213 Ki = 0.09 nM T48268 CX1OZ0 137637541 Ki = 0.23 nM T48268 CK0QM8 137637884 EC50 = 1 nM T48268 CT6EV9 137639112 Ki = 0.2 nM T48268 CV5QE0 137640407 Ki = 0.5 nM T48268 C6FPB9 137640743 Ki = 22 nM T48268 CK4I2U 137641357 Ki = 0.3 nM T48268 C0S6VY 137642160 Ki = 0.03 nM T48268 CUT89N 137644121 Ki = 3.8 nM T48268 C4Y3XB 137645530 Ki = 0.3 nM T48268 CAF5K6 137645887 Ki = 1 nM T48268 CEQG70 137646628 Ki = 250 nM T48268 C3U5GH 137647756 Ki = 0.09 nM T48268 CRS5I9 137648419 Ki = 0.22 nM T48268 CL8W1O 137650611 Ki = 0.3 nM T48268 C19KPO 137650826 Ki = 0.4 nM T48268 CQDC47 137653199 EC50 = 10 nM T48268 C5ST3G 137655126 Ki = 430 nM T48268 CRF49O 137655238 Ki = 0.1 nM T48268 CN51KY 137655435 Ki = 4 nM T48268 CH4EL7 137655489 Ki = 40 nM T48268 CU74BT 137656715 Ki = 47 nM T48268 CQZ1T6 137656978 Ki = 6 nM T48268 COG2K4 137657824 Ki = 550 nM T48268 CZFQ41 137660180 Ki = 26 nM T48268 C5TEM2 137660333 Ki = 0.2 nM T48268 CJE60O 137660726 Ki = 1 nM T48268 CDV21J 137661786 Ki = 6 nM T48268 CAP26G 139030523 EC50 = 540 nM T48268 COD7T0 145963877 Ki = 33.11 nM T48268 COZ43N 145964105 Ki = 44.67 nM T48268 CF0BH4 145965883 Ki = 398.11 nM T48268 CSN71J 145966403 Ki = 53.7 nM T48268 CUM9C5 145966622 Ki = 1.698 nM T48268 C5U7FM 145968467 Ki = 331.13 nM T48268 C2VK6W 145969866 Ki = 15.49 nM T48268 C26RKN 145971624 Ki = 19.05 nM T48268 C0N8ZF 145972981 Ki = 4.571 nM T48268 C6VB5Z 145974583 Ki = 12882.5 nM T48268 CZC60H 145975938 Ki = 26.92 nM T48268 CQ2Z7C 145976009 Ki = 6.31 nM T48268 C5YP8W 145976375 Ki = 295.12 nM T48268 CQAB74 145977894 Ki = 602.56 nM T48268 CC95GZ 145978811 Ki = 32.36 nM T48268 C6RV3M 145979282 Ki = 0.1 nM T48268 CUM97N 145979585 Ki = 0.4 nM T48268 CV8K7E 145979689 Ki = 0.2 nM T48268 CM7D2G 145981162 Ki = 0.1 nM T48268 C1YJ0P 145981769 Ki = 0.2 nM T48268 CH5A3J 145982070 Ki = 0.1 nM T48268 C9R8FK 145982167 Ki = 0.1 nM T48268 C6I5AL 145982333 Ki = 0.07 nM T48268 CO7R2A 145983175 Ki = 2 nM T48268 CF8T9A 145983929 Ki = 0.8 nM T48268 CM2C9Z 145986330 Ki = 0.4 nM T48268 C7VJ9I 145986532 Ki = 0.2 nM T48268 C3D6RX 145986700 EC50 = 2 nM T48268 C7U2SG 145987794 Ki = 0.1 nM T48268 C7C6XZ 145988269 Ki = 0.2 nM T48268 CC83DQ 145988741 Ki = 0.1 nM T48268 C5Q8HG 145988801 Ki = 2 nM T48268 CH04CY 145990308 Ki = 3 nM T48268 CRH4A6 145990662 Ki = 0.3 nM T48268 C2NF4G 145991111 Ki = 0.4 nM T48268 C73PGR 145991966 Ki = 0.4 nM T48268 CU94SI 145992795 Ki = 0.3 nM T48268 CX8HD4 145993188 Ki = 0.2 nM T48268 CZLY96 145993214 Ki = 0.2 nM T48268 C43VNT 145993566 Ki = 0.2 nM T48268 D01LAU 4284525 IC50 = 4000 nM T48268 D01SNS 4172142 Ki = 0.05 nM T48268 D01UIY 46885284 Ki = 1.59 nM T48268 D03AJW 44349108 Ki = 3.7 nM T48268 D03NND 22718564 Ki = 1.8 nM T48268 D03OGA 71533431 Ki = 0.07 nM T48268 D04BLO 57381112 Ki = 0.85 nM T48268 D04VGL 3976006 Ki = 0.01585 nM T48268 D05EDR 11630146 Ki = 2.94 nM T48268 D05TRX 22718561 Ki = 2.3 nM T48268 D05WKI 10244841 Ki = 0.16 nM T48268 D06AUM 9806449 Ki = 72.7 nM T48268 D07BKH 9798456 Ki = 0.36 nM T48268 D07EOD 22133318 Ki = 0.27 nM T48268 D07MFG 9957516 Ki = 51.3 nM T48268 D07YFL 24954989 Ki = 0.42 nM T48268 D07ZQU 46884598 Ki = 12.6 nM T48268 D08SGV 10849065 Ki = 75.86 nM T48268 D08TBF 71508234 EC50 = 0.24 nM T48268 D09ETU 46885285 Ki = 2.12 nM T48268 D09LPG 44208891 Ki = 0.8 nM T48268 D0B8PD 1858 Ki = 0.2 nM T48268 D0C5XQ 1832 Ki = 16 nM T48268 D0D6IK 10104923 Ki = 7.07 nM T48268 D0F6CD 5202 Ki > 100000 nM T48268 D0F6VI 46885230 Ki = 46.2 nM T48268 D0H6YF 115348 Ki = 0.15 nM T48268 D0I4DJ 24763223 Ki = 91 nM T48268 D0K1HD 24750192 Ki = 0.6457 nM T48268 D0L9YA 22718532 Ki = 4.3 nM T48268 D0O2GK 10059864 Ki = 0.34 nM T48268 D0OY8Y 11185529 Ki = 0.6607 nM T48268 D0Q0LH 9998187 Ki = 0.25 nM T48268 D0Q6HT 11536239 Ki = 2.75 nM T48268 D0R5JD 9870523 Ki = 112 nM T48268 D0RF4L 129776 Ki = 0.25 nM T48268 D0S3NS 25210130 Ki = 1.1 nM T48268 D0S6SN 1864 Ki = 5.5 nM T48268 D0TM0N 24749950 Ki = 27.54 nM T48268 D0U8OS 10750842 Ki = 0.751 nM T48268 D0V7VF 16094584 Ki = 0.2188 nM T48268 D0W7ZB 46885283 Ki = 26.1 nM T48268 D0WE4C 5311198 Ki = 0.5 nM T48268 D0Y2JY 53238181 Ki = 0.012 nM T79961 D01AZG 5073 Ki > 1000 nM T79961 D06HLY 5910 Ki = 10232.93 nM T79961 D08CTT 21855 Ki = 794.33 nM T79961 D0BZ7W 443879 Ki = 2.2 nM T79961 D0H3HM 60795 Ki > 1000 nM T79961 D0H7KF 5002 Ki > 1000 nM T79961 D0L4YD 154059 Ki = 43.65 nM T79961 D0M0AM 11693 IC50 = 0.1995 nM T79961 D0M6VK 71183 Ki = 0.2089 nM T79961 D0Q9HF 187 EC50 = 1.2 nM T79961 D0RD5W 154417 Ki = 0.14 nM T79961 D0RG3O 174174 Ki = 0.21 nM T79961 D0T0LM 4848 Ki = 35.48 nM T79961 D0U7BW 5831 EC50 = 360 nM T79961 D0V4QS 135398745 Ki = 10 nM T79961 D0VP1V 11434515 IC50 = 0.1585 nM T79961 D0Y5AM 444031 Ki = 2.3 nM T79961 D0Z1RV 135398737 Ki = 100 nM T79961 D07EFM 2230 EC50 = 600 nM T79961 D0I5XU 16065403 Ki = 0.169 nM T79961 D0K4HW 135409468 Ki = 51 nM T79961 D0N1HW 5311200 Ki > 10000 nM T79961 D02JNY 10030021 Ki = 316.23 nM T79961 D02KLW 180081 IC50 = 2 nM T79961 D06ACX 6436265 Ki = 489.78 nM T79961 D06DZI 107780 Ki > 10000 nM T79961 D08YVT 9894173 Ki = 85 nM T79961 D09FYQ 9577995 EC50 = 123 nM T79961 D0J8UV 9928284 EC50 = 1000 nM T79961 D0R1VL 132712 Ki = 1445.44 nM T79961 D0UX0T 9571002 Ki = 3162.28 nM T79961 D0VZ3D 129989 Ki = 831.76 nM T79961 CKD46H 4022 Ki = 3801.89 nM T79961 C7VMZ3 4108 Ki = 313 nM T79961 C2AF8D 6060 EC50 = 790 nM T79961 C5H9CN 9287 Ki > 10000 nM T79961 CV42HF 16817 EC50 = 1300 nM T79961 CNZD18 36381 Ki = 1161 nM T79961 CRCD50 60809 Ki = 9.333 nM T79961 C8E9XD 66007 IC50 = 10.3 nM T79961 CT0GD8 66266 Ki = 1288.25 nM T79961 C3WKC6 68835 IC50 = 71000 nM T79961 C3S8RF 71792 EC50 = 422 nM T79961 CA3W0P 100826 IC50 = 63000 nM T79961 C09JTU 199798 Ki = 2691 nM T79961 CC56KR 639794 Ki = 26915.35 nM T79961 C91GCI 657308 Ki = 1.04 nM T79961 CEGR96 657346 Ki = 21877.62 nM T79961 C04XRI 657347 Ki = 21877.62 nM T79961 CUD48J 952858 IC50 > 10000 nM T79961 CZ6Q4Y 1090198 IC50 > 10000 nM T79961 C4O6ZA 1090202 IC50 = 2300 nM T79961 CWFV17 1392038 IC50 = 3500 nM T79961 CH5WR4 1421986 IC50 > 10000 nM T79961 CZQ1J8 2048702 EC50 > 30000 nM T79961 CPL49A 2157678 EC50 > 30000 nM T79961 C7ET2M 3156646 IC50 = 1300 nM T79961 CI7DF6 3675988 Ki = 16595.87 nM T79961 C1WS4O 3724239 IC50 = 2600 nM T79961 CYI1N9 3810205 IC50 = 6600 nM T79961 CX3S8T 4715419 Ki = 19054.61 nM T79961 C12BJA 4995951 Ki = 1819.7 nM T79961 CS71UA 5189681 IC50 = 3490 nM T79961 CR5LG3 5310989 IC50 = 5999.2 nM T79961 C07PJQ 6603753 Ki = 13182.57 nM T79961 CFN7L4 6604866 Ki = 758.58 nM T79961 CWR31P 6861557 EC50 = 7600 nM T79961 CC8QT3 6891506 EC50 = 3000 nM T79961 C2IP0Y 7022778 Ki = 47863.01 nM T79961 CVSC58 7047822 Ki = 31622.78 nM T79961 C32TSZ 7141654 Ki = 138038.43 nM T79961 C7NJZ2 7141656 Ki = 15848.93 nM T79961 C7MBO3 9809330 Ki = 63.1 nM T79961 CTAC24 9885114 Ki = 964 nM T79961 CJ5K1D 9889312 Ki = 308.6 nM T79961 CUN81Q 9905249 Ki > 10000 nM T79961 C2U5LK 9905467 IC50 = 115.4 nM T79961 CYWQ50 9906447 Ki = 437 nM T79961 CDB9E1 9909907 Ki = 125.89 nM T79961 CXAV92 9911615 Ki = 1698.24 nM T79961 CXAY37 9913341 Ki = 398.11 nM T79961 CRV17M 9931930 Ki = 2238.72 nM T79961 C50NSR 9936450 Ki = 3.981 nM T79961 CCM72P 9974222 IC50 = 78.1 nM T79961 C9FR0C 9998508 Ki = 1230.27 nM T79961 CV7R9F 10020040 Ki > 10000 nM T79961 CQZ0K4 10027177 EC50 > 50000 nM T79961 CBJ63D 10043954 Ki = 977.24 nM T79961 C9OQ2S 10066369 Ki = 2187.76 nM T79961 CI6SD7 10066972 Ki = 1047.13 nM T79961 CCO72H 10082470 IC50 = 2100 nM T79961 C8NQ3I 10092649 Ki = 940 nM T79961 CG0O9Z 10109893 Ki = 3981.07 nM T79961 CUT05R 10114698 Ki = 5370.32 nM T79961 C90FZG 10139614 Ki > 28183.83 nM T79961 C0PO3J 10142923 Ki = 398.11 nM T79961 CG78WP 10160073 Ki = 11220 nM T79961 CZ8E9X 10160219 Ki = 2398.83 nM T79961 C1N4VJ 10182489 EC50 = 1258.93 nM T79961 COR14Y 10203251 Ki = 3388.44 nM T79961 C04QCB 10225881 Ki = 1479.11 nM T79961 C6A5KD 10226456 Ki = 630.96 nM T79961 CO64WJ 10236758 Ki = 5370.32 nM T79961 C3QGA5 10251795 EC50 > 50000 nM T79961 CW90FO 10261985 EC50 = 950 nM T79961 C1FCP7 10262466 Ki = 510 nM T79961 CH31DX 10267394 Ki > 10000 nM T79961 CC6RP7 10267601 IC50 = 54.1 nM T79961 CY3E5J 10274019 Ki = 1.66 nM T79961 CU89JD 10314060 Ki > 10000 nM T79961 C6S7GK 10354348 IC50 = 100000 nM T79961 C7BZ1R 10358345 IC50 = 138.9 nM T79961 C2B0IU 10421236 Ki > 10000 nM T79961 C5BEJ0 10442081 EC50 = 4700 nM T79961 CIRS06 10442337 EC50 = 2100 nM T79961 CC9AV4 10465280 EC50 = 110 nM T79961 CEF2O6 10478367 Ki > 10000 nM T79961 C8COH6 10499832 IC50 = 1567.9 nM T79961 CP9M5J 10516408 IC50 = 1127.9 nM T79961 C37PDA 10518821 IC50 = 31057 nM T79961 C6T1JW 10521205 IC50 = 159.2 nM T79961 C4WZ3R 10522202 IC50 = 1260.5 nM T79961 C5MB2F 10522336 IC50 = 328.6 nM T79961 C0K9HN 10538337 IC50 = 16901.9 nM T79961 C3Y6JB 10546275 IC50 = 85.4 nM T79961 CI3GQ6 10547222 IC50 = 1114.8 nM T79961 C6XKZ9 10549581 IC50 = 3565.8 nM T79961 CFD40Z 10567192 IC50 = 63 nM T79961 C4AL8Q 10569816 IC50 = 190.3 nM T79961 CB37SH 10573693 IC50 = 3108.6 nM T79961 C71VMD 10591874 IC50 = 272.8 nM T79961 C94VUE 10592484 IC50 = 537.3 nM T79961 C51LBK 10593954 IC50 = 255.8 nM T79961 CH2QU8 10594386 IC50 = 10969.8 nM T79961 CY54RA 10595006 Ki = 420 nM T79961 CZRJ60 10610375 IC50 = 977 nM T79961 CX01SE 10611310 IC50 = 1331.2 nM T79961 CO3H7D 10614695 IC50 = 1568.6 nM T79961 CJL4R1 10636001 IC50 = 602.9 nM T79961 C09XHV 10638050 IC50 = 374 nM T79961 C5VWL8 10641009 IC50 = 56.2 nM T79961 CONH15 10663572 IC50 = 42.5 nM T79961 C6WQ2Z 10664532 IC50 = 330.9 nM T79961 C8CF4H 10666533 IC50 = 499.7 nM T79961 C32KQX 10684720 IC50 = 254.9 nM T79961 C32EGP 10686988 IC50 = 222.1 nM T79961 C9O6LN 10688349 IC50 = 4264 nM T79961 CC21XD 10755732 IC50 = 264.7 nM T79961 CHL29Z 10755733 IC50 = 407.3 nM T79961 C4JXA3 10757736 IC50 = 1889.3 nM T79961 CPQ7Z3 10760249 IC50 = 24.8 nM T79961 C5P3DQ 10761219 IC50 = 5000 nM T79961 CX4LT3 10777692 IC50 = 4169.5 nM T79961 CA4QI2 10782321 IC50 = 2075.4 nM T79961 C4N9IT 10782462 IC50 = 214.5 nM T79961 C6FC0M 10784004 IC50 = 479.4 nM T79961 CV8TE0 10785471 IC50 = 235.6 nM T79961 C9SEA6 10806268 IC50 = 194.2 nM T79961 CGR64V 10808719 IC50 = 842 nM T79961 CK1D3J 10827157 IC50 = 558.9 nM T79961 CR1X5L 10829928 IC50 = 1467.3 nM T79961 CB7E2O 10846833 IC50 = 23000 nM T79961 CH9WK6 10851853 IC50 = 341.9 nM T79961 CX6AP3 10852843 IC50 = 2971.4 nM T79961 C5PRT6 10854879 IC50 = 400.6 nM T79961 C8HI5L 10854880 IC50 = 57.9 nM T79961 CZ85AJ 10862395 Ki = 3090.3 nM T79961 CHE9P4 10865439 Ki = 183 nM T79961 CCM3L9 10870954 Ki = 45708.82 nM T79961 C2YNC5 10871551 Ki = 776.25 nM T79961 CFAD04 10874119 Ki = 1122.02 nM T79961 CTV95B 10880435 Ki = 3630.78 nM T79961 C4A8QE 10916286 Ki = 4786.3 nM T79961 CQLR32 10919522 Ki = 150 nM T79961 CC12TE 10925451 Ki = 912.01 nM T79961 CU09AV 10937901 IC50 = 1910 nM T79961 CR7UE3 10946670 EC50 = 3190 nM T79961 C5LVY0 10949838 Ki = 3090.3 nM T79961 CE05FM 10951142 Ki = 478.63 nM T79961 C3K6JV 10957754 Ki = 3235.94 nM T79961 CN4QT5 10963509 Ki = 105 nM T79961 C4WV8L 10969390 Ki = 1995.26 nM T79961 CTYZ13 10969696 Ki = 2691.53 nM T79961 C41PXY 10982070 Ki = 3630.78 nM T79961 C9E2MP 10984804 Ki > 5000 nM T79961 C2W3GM 11000399 Ki = 10232.93 nM T79961 C6NH9T 11001809 Ki = 11220.18 nM T79961 CQ8D4K 11004046 Ki = 3715.35 nM T79961 C6BG1N 11006792 Ki = 2000 nM T79961 CU4Z0J 11011332 Ki = 7943.28 nM T79961 CZK86F 11011757 Ki = 309.03 nM T79961 CVA6U9 11012653 Ki = 2187.76 nM T79961 CPM1Z7 11012712 Ki = 6025.6 nM T79961 CW23BJ 11013666 Ki = 66.07 nM T79961 C6TF5I 11015312 Ki = 2511.89 nM T79961 C7Y1DO 11024241 Ki = 3235.94 nM T79961 C3L9ON 11034265 Ki = 1047.13 nM T79961 CHDT49 11039424 Ki = 37 nM T79961 CP9OJ6 11045444 Ki = 302 nM T79961 C4ZUH9 11048067 Ki = 2511.89 nM T79961 CR7W9T 11056389 EC50 = 7130 nM T79961 CQ8O3Y 11057942 Ki > 28183.83 nM T79961 CIG31V 11061341 Ki = 58 nM T79961 CT3XN5 11071537 Ki = 158.49 nM T79961 C5VQ6H 11079969 Ki = 2238.72 nM T79961 CWS56C 11092603 Ki = 501.19 nM T79961 C02MPO 11099206 Ki = 1995.26 nM T79961 CSNA03 11101362 Ki = 5370.32 nM T79961 CF81CB 11110049 Ki = 41686.94 nM T79961 C7ROJ1 11112362 Ki = 1122.02 nM T79961 C9CY0M 11120347 Ki = 1445.44 nM T79961 C2C4AN 11131099 Ki = 8912.51 nM T79961 C1T9WI 11143997 Ki = 1949.84 nM T79961 C10UKO 11189004 IC50 > 10000 nM T79961 C9FNM4 11431811 Ki = 0.0266 nM T79961 CGCF61 11515738 Ki < 100000 nM T79961 CY63VP 11523050 Ki = 33884.42 nM T79961 C07AJD 11530306 Ki = 57543.99 nM T79961 CWUP85 11542982 Ki < 100000 nM T79961 C6D1MA 11584660 IC50 = 630.96 nM T79961 CEHP14 11586481 Ki < 100000 nM T79961 CP3Y7J 11588240 Ki < 100000 nM T79961 CQ5PI4 11622544 Ki < 100000 nM T79961 CF2ZC0 11651360 Ki < 100000 nM T79961 CHKN81 11653111 Ki < 100000 nM T79961 C27XOS 11660220 Ki < 100000 nM T79961 C0N4BQ 11672895 Ki < 100000 nM T79961 CN4Z5C 11679149 IC50 > 10000 nM T79961 CW8CE2 11694118 Ki < 100000 nM T79961 CF8MO2 11694119 Ki < 100000 nM T79961 C9BF1S 11715398 Ki < 100000 nM T79961 CEY7J3 11729182 Ki = 19498.45 nM T79961 CPG15O 11743399 IC50 > 1000 nM T79961 C4QVR6 11748799 Ki = 371.54 nM T79961 CQLP36 11759058 Ki = 66069.34 nM T79961 CW3GA7 11759212 Ki = 724.44 nM T79961 CBM05D 11759379 Ki = 2344.23 nM T79961 CFZ4L5 11767229 Ki = 210 nM T79961 C39HRB 11793999 IC50 = 472.2 nM T79961 CT4F2C 11808040 Ki = 87.1 nM T79961 CXQ10I 11808946 Ki = 676.08 nM T79961 C6EXD3 11808947 Ki = 1122.02 nM T79961 C30WRH 11809446 Ki = 17378.01 nM T79961 CQW16Z 11819782 Ki = 52480.75 nM T79961 CJIA51 11828362 Ki = 30 nM T79961 CR9FJ2 11833737 Ki = 5888.44 nM T79961 CZ3AX9 11834199 Ki = 2089.3 nM T79961 C8JQL7 11957735 IC50 > 10000 nM T79961 CL91TM 11968014 Ki = 1.288 nM T79961 CYU4P5 12739458 Ki = 6546 nM T79961 C12KIW 13248082 EC50 = 4660 nM T79961 CR10FQ 13567080 Ki = 2.818 nM T79961 CA87RQ 14660293 IC50 = 100000 nM T79961 CMO81H 14925759 Ki = 27542.29 nM T79961 C7VAI1 15011772 IC50 > 10000 nM T79961 CVNK57 15065550 Ki = 51.29 nM T79961 CO4P1Q 16001212 EC50 > 10000 nM T79961 CUB5X2 16038385 EC50 > 10000 nM T79961 CZ47FJ 16071018 EC50 = 794.33 nM T79961 C3T0UX 16085999 Ki = 1700 nM T79961 CWI32N 16086000 Ki = 1600 nM T79961 C71HBL 16086001 Ki = 1600 nM T79961 C7EM1G 16086003 Ki > 5100 nM T79961 CFU72Z 16086004 Ki > 5100 nM T79961 CTOM27 16086005 Ki = 950 nM T79961 C7WF9Y 16086059 Ki = 3500 nM T79961 C05YVJ 16086060 Ki = 1700 nM T79961 CMQ8U3 16086061 Ki = 2800 nM T79961 CEI8G1 16086062 Ki = 3100 nM T79961 CGB89M 16086063 Ki = 940 nM T79961 CUS73E 16086064 Ki = 3200 nM T79961 CHJ07L 16086065 Ki > 5100 nM T79961 CEV68D 16086066 Ki = 2500 nM T79961 CIX9M7 16086067 Ki = 2700 nM T79961 C1XZ7V 16094783 Ki = 251.19 nM T79961 CO16DS 16094788 Ki = 100 nM T79961 CYN71L 16094791 Ki = 630.96 nM T79961 C2HK7W 16094793 Ki = 251.19 nM T79961 C9R0JN 16094810 Ki = 100 nM T79961 CTYI57 16115796 Ki = 3.236 nM T79961 C5HSD9 16115797 Ki = 1.995 nM T79961 CQ85FK 16115798 Ki = 1.995 nM T79961 CR1Z4N 16115799 Ki = 1.202 nM T79961 CLA6E0 16115800 Ki = 3.467 nM T79961 CTE0R7 16115942 Ki = 3.236 nM T79961 C7IC9E 16115944 Ki = 0.1995 nM T79961 CQ3C9X 16115946 Ki = 0.7762 nM T79961 C0JGY1 16115950 Ki = 5.623 nM T79961 CZ67DO 16115951 Ki = 1.349 nM T79961 CO3YU4 16116082 Ki = 0.4074 nM T79961 C3IKJ0 16116084 Ki = 0.1072 nM T79961 CWU6P3 16123945 EC50 = 1258.93 nM T79961 CZ2IS9 16660294 Ki > 10000 nM T79961 CDB83R 17516658 EC50 = 10000 nM T79961 C7T8JC 19958494 Ki > 10000 nM T79961 C6LI5E 19958507 Ki > 10000 nM T79961 C3T5HF 21509921 Ki = 5128.61 nM T79961 CBN84K 22065997 Ki > 10000 nM T79961 C5WCD3 22745278 EC50 = 34.3 nM T79961 CMLE80 22772867 IC50 > 10000 nM T79961 C5Y1MK 23983764 Ki = 6.166 nM T79961 CY21RE 24841480 Ki = 6 nM T79961 CF26NI 24865894 Ki = 4570.88 nM T79961 CJ4FM6 24865895 Ki = 3715.35 nM T79961 C9YN3A 24894514 Ki = 63095.73 nM T79961 C8ND1U 24894515 Ki = 75857.76 nM T79961 CX2HR8 24894516 Ki = 39810.72 nM T79961 CG4B9R 24894624 Ki = 20892.96 nM T79961 C7KF9R 24894626 Ki = 3630.78 nM T79961 CFA60S 24894627 Ki = 3162.28 nM T79961 CT8B3K 24894629 Ki = 4677.35 nM T79961 CMF04K 24894631 Ki = 44668.36 nM T79961 CP08SJ 24894632 Ki = 21877.62 nM T79961 CLJK58 24894633 Ki = 31622.78 nM T79961 CR86FA 24894634 Ki = 23442.29 nM T79961 C9J3NX 24894636 Ki = 9549.93 nM T79961 CR7D1L 24967746 EC50 = 12.59 nM T79961 C5MYC3 25010776 EC50 > 30000 nM T79961 CA20NZ 25025581 Ki = 100 nM T79961 CBY3O2 25070582 IC50 = 300 nM T79961 CXBF68 25110764 EC50 > 50000 nM T79961 C50IKG 25110765 EC50 > 50000 nM T79961 CE2OG1 25199525 EC50 = 1000 nM T79961 CRFJ43 25207745 EC50 = 1000 nM T79961 CP2T6G 25230693 EC50 = 158.49 nM T79961 CJ7F2P 26415263 EC50 = 6165.95 nM T79961 C1PVI6 26415265 EC50 = 3300 nM T79961 CS69PF 30855719 EC50 > 10000 nM T79961 C45ZNS 42596928 Ki = 4.365 nM T79961 C5DC7E 42598357 EC50 = 398.11 nM T79961 CO6QB0 42598358 EC50 = 50.12 nM T79961 CDPA93 42598359 EC50 = 1258.93 nM T79961 CAM5P6 42598360 EC50 = 158.49 nM T79961 C58SRK 42598586 EC50 = 5011.87 nM T79961 CYL45Z 42598591 EC50 = 19.95 nM T79961 C6S2HI 42598828 EC50 = 158.49 nM T79961 C2GYA4 42598829 EC50 = 398.11 nM T79961 C5CZ7P 42599068 EC50 = 125.89 nM T79961 C7O2ZV 42599070 EC50 = 19.95 nM T79961 C6BUZ5 42599071 EC50 = 316.23 nM T79961 C5N1OM 44157160 EC50 = 1930 nM T79961 C8U6FX 44157241 EC50 = 3960 nM T79961 CF2EB6 44157243 EC50 = 1860 nM T79961 CH8LP5 44157319 EC50 > 10000 nM T79961 CL1QC4 44157714 EC50 = 4070 nM T79961 C8V2AP 44158003 EC50 = 3280 nM T79961 C0L3XT 44158005 EC50 = 7150 nM T79961 CNK83R 44158075 EC50 = 1700 nM T79961 CQ1EY4 44158077 EC50 = 4090 nM T79961 CV20NI 44158078 EC50 > 30000 nM T79961 C5NJ4W 44158139 EC50 = 3260 nM T79961 C3ABS1 44158142 EC50 = 2100 nM T79961 CAK93Y 44158221 EC50 = 1850 nM T79961 CMR7T1 44204999 EC50 = 1584.89 nM T79961 C6GXL0 44208359 EC50 = 1200 nM T79961 CGR6J0 44251556 EC50 = 600 nM T79961 C2K0VZ 44253016 EC50 > 10000 nM T79961 C2LFH7 44274302 Ki = 17782.79 nM T79961 CZX4M3 44274317 Ki = 54954.09 nM T79961 C5L3FV 44274400 Ki = 66069.34 nM T79961 CF47ZS 44274417 Ki = 52480.75 nM T79961 CCK63Z 44274432 Ki = 53703.18 nM T79961 CZ1U0E 44274433 Ki = 53703.18 nM T79961 C3XP7C 44274441 Ki = 30199.52 nM T79961 CO1RL0 44274468 Ki = 26915.35 nM T79961 C9JX7D 44274469 Ki = 19054.61 nM T79961 CF36IC 44274477 Ki = 54954.09 nM T79961 CC2OD4 44278111 Ki > 10000 nM T79961 CRMA84 44278114 Ki > 10000 nM T79961 CF0Y4M 44278115 Ki > 10000 nM T79961 C9TWN3 44302727 IC50 = 8211.3 nM T79961 C5S8UL 44302728 IC50 = 26644.8 nM T79961 CQ4B5T 44302741 IC50 = 3807.6 nM T79961 C0AZF5 44302755 IC50 = 47361.5 nM T79961 CR5T1J 44302775 IC50 = 8624 nM T79961 CY8PD1 44302776 IC50 = 3884.2 nM T79961 C7GY5J 44302788 IC50 = 4093 nM T79961 CAV72D 44302793 IC50 = 43462.7 nM T79961 CV9QM6 44302813 IC50 = 4187.1 nM T79961 C43QTF 44302833 IC50 = 1731.8 nM T79961 CF74EQ 44302834 IC50 = 2033.9 nM T79961 C6J3EY 44302879 IC50 = 5760.1 nM T79961 CIU20B 44302900 IC50 = 4737 nM T79961 CGNA91 44302901 IC50 = 17980.7 nM T79961 CSK4B0 44346542 IC50 = 508.2 nM T79961 C7YTV9 44385809 Ki = 1100 nM T79961 CHD9O7 44386115 Ki = 200 nM T79961 C1B4QL 44403095 Ki > 10000 nM T79961 C1YL7Z 44403098 Ki > 10000 nM T79961 CFV98A 44403101 Ki > 10000 nM T79961 C6OY9S 44403102 Ki > 10000 nM T79961 CH4SX6 44403105 Ki > 10000 nM T79961 C12FIH 44403106 Ki > 10000 nM T79961 C4LKC1 44404394 Ki > 10000 nM T79961 C3EJ4G 44404396 Ki > 10000 nM T79961 C6GLV1 44408714 Ki = 3801.89 nM T79961 C4QTI3 44415886 Ki > 5400 nM T79961 CC9AV3 44418764 Ki = 251.19 nM T79961 CV6UQ3 44419370 Ki > 100000 nM T79961 C2N5LX 44422691 Ki = 7762.47 nM T79961 CIRB78 44422696 Ki = 30199.52 nM T79961 CHT24X 44422698 Ki = 44668.36 nM T79961 CDE8A1 44428745 Ki = 169.82 nM T79961 CG45PO 44437242 Ki = 6310 nM T79961 C6I2JO 44437248 Ki = 7514 nM T79961 CZI05O 44437258 Ki = 1836 nM T79961 C2DAH1 44437265 Ki > 10000 nM T79961 C2EFY1 44437274 Ki > 10000 nM T79961 CXD1P2 44437278 Ki > 10000 nM T79961 C3E5FV 44437285 Ki > 10000 nM T79961 C7VP1Y 44437297 Ki = 4116 nM T79961 C5GT7C 44437302 Ki > 10000 nM T79961 C37QFT 44437307 Ki = 5664 nM T79961 C36LXN 44446840 Ki = 67608.3 nM T79961 C6S4XU 44448379 Ki = 25703.96 nM T79961 C0ZLX8 44448383 Ki = 588.84 nM T79961 C1USW7 44448418 Ki = 7585.78 nM T79961 C8NB9P 44448421 Ki = 776.25 nM T79961 CMF5E6 44448456 Ki = 18197.01 nM T79961 CH9IC4 44448495 Ki = 6918.31 nM T79961 CHAX49 44448499 Ki = 1548.82 nM T79961 CA9QL5 44448537 Ki = 9549.93 nM T79961 CJK41H 44448645 Ki = 707.95 nM T79961 CR4ZT2 44450620 Ki = 24547.09 nM T79961 C5H7OQ 44450621 Ki = 23442.29 nM T79961 CZ50IM 44450622 Ki = 10715.19 nM T79961 CS5CD3 44450624 Ki = 10232.93 nM T79961 CFN4B5 44450637 Ki = 22908.68 nM T79961 C12XGE 44456400 Ki > 10000 nM T79961 CVA67X 44568347 Ki = 120 nM T79961 CY9C2A 44571572 Ki > 100000 nM T79961 CHUN40 44578928 EC50 > 50000 nM T79961 CZYP06 44578975 EC50 > 50000 nM T79961 CCIT12 44578976 EC50 > 50000 nM T79961 CW53ZF 44578977 EC50 > 50000 nM T79961 CYHM34 44578978 EC50 > 50000 nM T79961 CGF7A4 44579375 EC50 > 50000 nM T79961 C1OCB6 44579416 EC50 > 50000 nM T79961 CARW17 44579417 EC50 > 50000 nM T79961 C2DFV7 44579418 EC50 > 50000 nM T79961 CTC8H6 44579419 EC50 > 50000 nM T79961 CYR0O3 44579457 EC50 > 50000 nM T79961 CF1EA4 44579458 EC50 > 50000 nM T79961 CQ4Y8O 44589531 EC50 > 30000 nM T79961 CL40CM 44589593 EC50 > 30000 nM T79961 CKS5V4 44589594 EC50 > 30000 nM T79961 CXB30W 44589595 EC50 > 30000 nM T79961 CM5LJ8 44589596 EC50 > 30000 nM T79961 CPXE19 44589643 EC50 > 30000 nM T79961 C8AJO6 44589644 EC50 > 30000 nM T79961 CFS1A4 44589645 EC50 > 30000 nM T79961 C71EHI 44589646 EC50 > 30000 nM T79961 CQB5A9 44589681 EC50 = 34.3 nM T79961 CUA62X 44593616 Ki = 338.84 nM T79961 CN9ID8 44593617 Ki = 229.09 nM T79961 CDM56I 44593618 Ki = 58.88 nM T79961 CU63PQ 44593619 Ki = 25.12 nM T79961 CL8D2S 44593620 Ki = 30.2 nM T79961 CI97KQ 44593621 Ki = 380.19 nM T79961 CL5O8E 44602489 EC50 = 1900 nM T79961 CH2Z3O 44610056 Ki = 1.1 nM T79961 CVZ6Y1 44627739 Ki = 97.72 nM T79961 CE6A9F 44627740 Ki = 7.079 nM T79961 C6EU7P 44627741 Ki = 104.71 nM T79961 CW40TR 44627742 Ki = 54.95 nM T79961 C5GIU6 44627743 Ki = 37.15 nM T79961 CK9DO1 44627745 Ki = 11.48 nM T79961 CJ8S1L 44627747 Ki = 31.62 nM T79961 C5LY8C 44627851 Ki = 15.49 nM T79961 CC4A3X 44627853 Ki = 3.311 nM T79961 CH4N5J 44627854 Ki = 27.54 nM T79961 CO8C6D 44627855 Ki = 467.74 nM T79961 COL8E1 44627856 Ki = 1548.82 nM T79961 C6WS7M 44627857 Ki = 1.549 nM T79961 C43BJY 44627859 Ki = 12.02 nM T79961 CW0X6A 44627955 Ki = 229.09 nM T79961 CXNF31 44627957 Ki = 870.96 nM T79961 C9U0VH 45259185 Ki = 181.97 nM T79961 CNC1R2 45259186 Ki = 30.2 nM T79961 CP2CZ7 45259187 Ki = 194.98 nM T79961 CW14TS 45259188 Ki = 3.02 nM T79961 CO8W1X 45259189 Ki = 14.13 nM T79961 CF16YZ 45259190 Ki = 41.69 nM T79961 C7L1CU 45266348 Ki = 141.25 nM T79961 CK8N4L 45266386 Ki = 33884.42 nM T79961 C98FDW 45281794 EC50 = 1600 nM T79961 CPJ3F6 45281796 EC50 = 3900 nM T79961 C2YJ8M 45281797 EC50 = 2800 nM T79961 C0Y1ER 45281798 EC50 = 4800 nM T79961 CWX07N 45281801 EC50 = 3600 nM T79961 CH0I4B 45281803 EC50 = 3300 nM T79961 CRX2U3 45281807 EC50 = 5700 nM T79961 C5FX7A 45281808 EC50 = 2700 nM T79961 CGA2Z8 45494871 EC50 > 10000 nM T79961 CU4V5R 46227410 Ki = 63095.73 nM T79961 CWQ1L9 46227412 Ki = 15488.17 nM T79961 CX2E6A 46227414 Ki > 100000 nM T79961 C0Z4RD 46227416 Ki > 100000 nM T79961 CK2R5G 46227454 Ki = 97723.72 nM T79961 C8OZI6 46227456 Ki = 28183.83 nM T79961 CB45NM 46227458 Ki > 100000 nM T79961 C1J0IF 46227460 Ki = 52480.75 nM T79961 CQ4DI6 46227480 Ki = 83176.38 nM T79961 CHKL80 46227482 Ki = 32359.37 nM T79961 CVP7T6 46227484 Ki = 16595.87 nM T79961 CC6RH5 46227486 Ki = 66069.34 nM T79961 CSQ0V3 46227554 Ki = 93325.43 nM T79961 CAY5R2 46438676 EC50 > 10000 nM T79961 CK1X9S 46830361 IC50 = 830 nM T79961 C1Q0MH 46830362 IC50 = 4100 nM T79961 CH3ID7 46830363 IC50 > 10000 nM T79961 C01YTE 46871665 IC50 = 5011.87 nM T79961 CUY51M 46871666 IC50 > 10000 nM T79961 CYLZ50 46871844 IC50 = 501.19 nM T79961 CCZ5I8 46883796 IC50 = 4100 nM T79961 CVCF68 46883843 IC50 > 10000 nM T79961 CW70YU 46890977 IC50 = 794.33 nM T79961 CJ74AZ 46891076 IC50 = 1584.89 nM T79961 CTSZ49 46891179 IC50 = 6309.57 nM T79961 COT8S4 46891375 EC50 > 10000 nM T79961 CW1YX7 46891488 IC50 > 10000 nM T79961 CB1Z5A 46905390 IC50 = 162.5 nM T79961 CMU06V 46945662 EC50 = 3800 nM T79961 C67XQI 46945663 EC50 = 1500 nM T79961 CKN3S0 46945664 EC50 = 3200 nM T79961 C8V7JF 46945864 EC50 = 2200 nM T79961 CM75JZ 46945865 EC50 = 2800 nM T79961 C7IAW9 49663949 IC50 < 1500 nM T79961 CD39WZ 49665121 IC50 = 5160 nM T79961 C2LZJ0 49783209 Ki = 972 nM T79961 C57SMG 49783415 Ki = 4058 nM T79961 C0TG6I 49783419 Ki > 10000 nM T79961 C2TAI1 49797319 Ki > 10000 nM T79961 C20SCO 49797320 Ki = 6885 nM T79961 C29QSB 49797322 Ki = 544 nM T79961 CHS34N 49797323 Ki > 10000 nM T79961 C9V5OK 49797324 Ki > 10000 nM T79961 CT4QU7 49797325 Ki = 5139 nM T79961 C1WG5X 49797326 Ki > 10000 nM T79961 C13SKB 49797327 Ki > 10000 nM T79961 CLB8A4 49797328 Ki > 10000 nM T79961 C7ROA4 49797387 Ki = 2884.03 nM T79961 CQX3I5 49797388 Ki = 831.76 nM T79961 C9VG5A 49797390 Ki = 229086.77 nM T79961 C6RES8 49797391 Ki = 23442.29 nM T79961 C2E0DY 49797392 Ki = 123026.88 nM T79961 CLF8X5 49797394 Ki = 13489.63 nM T79961 CXD65I 49797395 Ki = 1412.54 nM T79961 CPI6N0 49853777 IC50 > 100000 nM T79961 C94GDK 49853778 IC50 > 100000 nM T79961 CHV3U8 49853881 IC50 > 100000 nM T79961 CTBY97 49853883 IC50 = 74000 nM T79961 CQP63D 49853884 IC50 = 26000 nM T79961 CY8M9A 49853885 IC50 > 100000 nM T79961 CN0JU9 49853987 IC50 > 100000 nM T79961 C8DVX6 49855131 IC50 > 100000 nM T79961 C51INK 50841366 IC50 > 10000 nM T79961 C2RY0J 50878551 Ki > 10000 nM T79961 C1W6TV 50898777 Ki > 10000 nM T79961 CXMZ73 50898778 Ki > 10000 nM T79961 CE4KP1 51050257 Ki > 10000 nM T79961 CM47HJ 52176747 IC50 = 6500 nM T79961 C8XK0E 52940924 EC50 = 5900 nM T79961 C96TXG 52941424 EC50 = 3100 nM T79961 C0FER9 52941977 EC50 = 4400 nM T79961 C3LYF9 52943684 EC50 = 3200 nM T79961 C0FA2T 52944339 EC50 > 30000 nM T79961 C3GV7Z 52946099 EC50 > 30000 nM T79961 CT4RA5 52946135 EC50 > 30000 nM T79961 CU79HQ 52947398 EC50 = 1600 nM T79961 C10AGJ 52947457 EC50 = 2100 nM T79961 CSFM86 52948724 EC50 > 30000 nM T79961 C3AXD0 52949292 EC50 = 4000 nM T79961 C2G3UC 52949811 EC50 > 30000 nM T79961 CC3B5V 52949833 EC50 = 2800 nM T79961 CUR7D0 52950176 EC50 = 2400 nM T79961 C6KU3Z 53303986 IC50 = 4900 nM T79961 CR4W9L 53324553 Ki = 1827 nM T79961 CG24AT 53381002 IC50 > 10000 nM T79961 CS1OI7 53382523 EC50 > 30000 nM T79961 CWR16G 53382542 EC50 > 30000 nM T79961 CVXH19 53384880 EC50 = 33 nM T79961 C7YP3A 53385782 EC50 = 3700 nM T79961 CPGC12 53385783 EC50 > 10000 nM T79961 CMOZ61 53475319 Ki = 2297 nM T79961 C8WHT5 56593934 Ki = 10000 nM T79961 CH37LU 56663451 Ki = 7036 nM T79961 CU0NE5 56672197 Ki = 5484 nM T79961 C9IH2R 56764681 IC50 > 10000 nM T79961 CD83PO 56764696 IC50 > 10000 nM T79961 CB0P9N 56944383 Ki > 1000 nM T79961 C1TC7Q 56963799 Ki = 336 nM T79961 C3WC7Z 56965018 Ki = 5.37 nM T79961 CUP4Y0 57326139 Ki = 26302.68 nM T79961 C1G9XY 57326141 Ki > 100000 nM T79961 CG3YS9 57326143 Ki = 10232.93 nM T79961 CCYU25 57326145 Ki = 33113.11 nM T79961 CS86GL 57326232 Ki = 107.15 nM T79961 C3AF0Z 57326234 Ki = 1.698 nM T79961 CLSW35 57326236 Ki = 7585.78 nM T79961 CL3R5D 57326238 Ki = 31622.78 nM T79961 C4G1LB 57326325 Ki = 81.28 nM T79961 C6CB9J 57326326 Ki = 1.82 nM T79961 C5OJP0 57391102 EC50 > 30000 nM T79961 C17GMJ 57393065 IC50 > 30000 nM T79961 CER4F5 57525833 EC50 = 446.68 nM T79961 C27DQU 57525835 EC50 = 524.81 nM T79961 CL4G1K 57525851 EC50 = 2200 nM T79961 CW5QM8 57525858 EC50 = 588.84 nM T79961 CQ5BG6 57525860 EC50 = 407.38 nM T79961 CH83EP 57525867 EC50 = 1400 nM T79961 CI4CV5 57525872 EC50 = 1047.13 nM T79961 C9TMZ3 57558000 Ki > 100000 nM T79961 CA14SG 58653718 Ki > 100000 nM T79961 CN4C7D 59025695 IC50 = 2344.23 nM T79961 C6MQY2 59025917 IC50 = 1800 nM T79961 CJQ63V 59025979 IC50 = 2000 nM T79961 C6C7EJ 60138185 Ki = 30199.52 nM T79961 C8WGS2 60138186 Ki = 3981.07 nM T79961 CAZ9B3 62705488 IC50 > 10000 nM T79961 C9F4JW 62705832 IC50 > 10000 nM T79961 CA5FP7 66561966 Ki = 2665 nM T79961 C3XL7O 66561967 Ki = 802 nM T79961 CKD60A 70789640 Ki = 1749 nM T79961 C9VZ8J 71450550 Ki = 924 nM T79961 CY3M8B 71451570 IC50 = 82 nM T79961 C4NDR3 71452382 Ki = 1700 nM T79961 CYK20Z 71452384 Ki > 10000 nM T79961 CDTW09 71452387 Ki = 1555 nM T79961 C6G2HC 71455894 Ki = 4157 nM T79961 CVI7S2 71457690 Ki > 10000 nM T79961 CP7JI0 71457691 Ki = 931 nM T79961 CK5T4P 71459604 Ki > 10000 nM T79961 C2OIW1 71461631 IC50 = 96.8 nM T79961 C1Y9IC 71463063 Ki = 5813 nM T79961 C68UAI 71574174 Ki = 3340 nM T79961 CK3T7C 71574175 Ki > 100000 nM T79961 CBZ78V 71574176 Ki > 100000 nM T79961 C61VXZ 71574177 Ki > 100000 nM T79961 C5OQ7W 71574178 Ki > 100000 nM T79961 CI0HU8 71574179 Ki > 100000 nM T79961 C6U4XJ 71574180 Ki > 100000 nM T79961 C0ZDF2 71574268 Ki > 100000 nM T79961 C0R3KB 71574269 Ki > 100000 nM T79961 CJ4WU1 71574271 Ki > 100000 nM T79961 C8ORK4 71574275 Ki = 2620 nM T79961 CCA49H 71574365 Ki = 1140 nM T79961 CRT07Q 71574367 Ki > 100000 nM T79961 C0E9SQ 71575024 Ki = 1250 nM T79961 CJ3H1M 71575025 Ki = 150 nM T79961 CR04XZ 71575026 Ki = 3610 nM T79961 C3MJ7B 71575027 Ki = 470 nM T79961 C8XEB3 71575028 Ki > 100000 nM T79961 C0XWU1 71575029 Ki = 290 nM T79961 C09DIB 71575117 Ki = 190 nM T79961 CM5OX8 71575118 Ki = 410 nM T79961 CAS1M2 71575119 Ki = 370 nM T79961 CL3A8V 71575120 Ki = 440 nM T79961 CQ21RK 71575121 Ki > 100000 nM T79961 CN82HY 71575122 Ki = 230 nM T79961 CDAH09 71575123 Ki = 280 nM T79961 CZP59X 71575219 Ki = 120 nM T79961 CGR20T 71575220 Ki = 2460 nM T79961 C95ZSD 71575221 Ki > 100000 nM T79961 CTA7V5 71575222 Ki > 100000 nM T79961 CT03QG 71575223 Ki = 760 nM T79961 CYS85C 71575224 Ki = 140 nM T79961 C4I8TD 71575225 Ki = 190 nM T79961 CP3OI1 71575336 Ki > 100000 nM T79961 CQUT29 71575337 Ki = 30 nM T79961 CE4L0U 71575338 Ki > 100000 nM T79961 CJ5VK2 71575339 Ki > 100000 nM T79961 CY1Q9O 71575447 Ki = 60 nM T79961 CEX7R3 71575448 Ki > 100000 nM T79961 CD48AB 71575449 Ki > 100000 nM T79961 C0VAJ8 71575450 Ki = 1160 nM T79961 CD86FK 71575451 Ki > 100000 nM T79961 CVR1Q3 71575452 Ki = 630 nM T79961 CL3YP2 71575453 Ki = 190 nM T79961 CLX37P 71575548 Ki = 110 nM T79961 CHB4M1 71575549 Ki = 280 nM T79961 C3LE4R 71575550 Ki = 80 nM T79961 C93ZCM 71575551 Ki = 740 nM T79961 CNS4V8 71575552 Ki = 2240 nM T79961 CM9SQ2 71575553 Ki = 5040 nM T79961 CMTB67 71575554 Ki > 100000 nM T79961 C1XV6F 71575649 Ki = 3070 nM T79961 CKI50H 71575650 Ki = 2350 nM T79961 CTSL25 71575651 Ki > 100000 nM T79961 C89MPL 71575652 Ki = 740 nM T79961 COY38T 71575653 Ki = 2680 nM T79961 CK6F1D 71575654 Ki = 2410 nM T79961 CM8UN7 71598549 IC50 = 478.63 nM T79961 C0RNW1 71598550 IC50 > 30000 nM T79961 CR4MH1 71607051 IC50 = 4100 nM T79961 CO9IQ3 71607053 IC50 > 10000 nM T79961 C2ZVH7 71607056 IC50 = 790 nM T79961 C4T6JM 71607062 IC50 > 10000 nM T79961 CW3KS4 71607066 IC50 = 1380 nM T79961 C89PCR 71607067 IC50 = 2089.3 nM T79961 CW6UE5 71607070 IC50 > 10000 nM T79961 CL6H1Q 71607072 IC50 > 10000 nM T79961 CK6HT3 71607077 IC50 < 10000 nM T79961 CQ2G5K 71607080 IC50 = 3000 nM T79961 CTE7O0 71607082 IC50 > 10000 nM T79961 CEM57I 71607084 IC50 = 2300 nM T79961 C8J6DX 71607089 IC50 = 3019.95 nM T79961 C01IME 71607090 IC50 = 3467.37 nM T79961 C10KST 71607091 IC50 = 4466.84 nM T79961 CH1T5S 71607096 IC50 = 2600 nM T79961 C1OE9J 71607097 IC50 = 1047.13 nM T79961 C5O2XT 71607107 IC50 > 10000 nM T79961 CN1OQ7 71607111 IC50 = 3800 nM T79961 C4UZV5 71607115 IC50 > 10000 nM T79961 CI2U5L 71607117 IC50 = 1288.25 nM T79961 C9V7YQ 71607121 IC50 = 5750 nM T79961 C0F6KE 71607129 IC50 = 1949.84 nM T79961 CET7U2 71607130 IC50 = 1000 nM T79961 CINP32 71607135 IC50 > 10000 nM T79961 CE1IQ8 71607137 IC50 = 4897.79 nM T79961 C9I1TX 71717914 Ki > 100000 nM T79961 CWP9X6 71737574 EC50 = 3090.3 nM T79961 CO7K1B 71737578 EC50 = 1548.82 nM T79961 C1Y4QO 71737582 EC50 > 10000 nM T79961 C1Y7TQ 71737591 EC50 > 10000 nM T79961 CT8OL3 71737602 EC50 = 970 nM T79961 CC65ZW 71737606 EC50 = 2344.23 nM T79961 CWJ91H 71737611 EC50 = 1698.24 nM T79961 C5FNH2 71737612 EC50 > 10000 nM T79961 C8Q6XC 71737616 EC50 > 10000 nM T79961 CP64EY 71737617 EC50 = 740 nM T79961 CL5K6S 71737618 EC50 = 758.58 nM T79961 C4WO0I 71737619 EC50 = 930 nM T79961 CD47KT 71737624 EC50 = 724.44 nM T79961 C24NFO 71737625 EC50 > 10000 nM T79961 CXZ5M1 71737627 EC50 = 1500 nM T79961 C04BCG 71737628 EC50 = 1110 nM T79961 CYGE50 71737645 EC50 = 2600 nM T79961 C4D0PN 71737646 EC50 = 1600 nM T79961 C1J3KL 71737647 EC50 = 2100 nM T79961 C9FZA3 71737648 EC50 = 478.63 nM T79961 C2A4LN 71737675 EC50 = 640 nM T79961 CI1EV5 71737677 EC50 = 870 nM T79961 CPI6U4 71737681 EC50 = 870 nM T79961 CVWE38 71737683 EC50 = 5495.41 nM T79961 C5MF4L 71737709 EC50 = 346.74 nM T79961 COUY23 71737725 EC50 > 10000 nM T79961 CCW4A9 71737726 EC50 > 10000 nM T79961 C9S7IY 71737757 EC50 > 10000 nM T79961 CI8B3Q 71737760 EC50 = 7400 nM T79961 CU0D4K 71737763 EC50 = 750 nM T79961 CWI28G 71737767 EC50 > 10000 nM T79961 CMQA74 71737771 IC50 = 1300 nM T79961 CY2L8R 71771053 EC50 = 1800 nM T79961 CZIN07 71771054 EC50 = 2951.21 nM T79961 CG6WC9 71771056 EC50 = 1258.93 nM T79961 CW5NO7 71771057 EC50 > 10000 nM T79961 C43UNK 71771058 EC50 = 154.88 nM T79961 C3FQY2 71806339 IC50 = 660.69 nM T79961 C7DTQ3 71806933 IC50 > 10000 nM T79961 CHE5O6 72545089 Ki > 100000 nM T79961 CI6D4E 72545091 Ki > 100000 nM T79961 CKFW54 72545094 Ki > 100000 nM T79961 CWLO54 72545096 Ki > 100000 nM T79961 C5D4PA 72545098 Ki > 100000 nM T79961 CR39AG 72545326 Ki > 100000 nM T79961 C5HLF7 72545329 Ki > 100000 nM T79961 CC65OA 73213195 Ki > 10000 nM T79961 CW83DK 73213196 Ki > 10000 nM T79961 CK0HR9 73346334 Ki = 2001 nM T79961 C6J0TM 73346336 Ki = 2907 nM T79961 CY60RD 73347826 Ki = 5801 nM T79961 CC35AI 73347827 Ki = 4243 nM T79961 C58SJG 73349591 Ki > 100000 nM T79961 CA6Z1P 73349592 Ki > 100000 nM T79961 CDS4F1 73350931 Ki = 1987 nM T79961 CA8L9Y 73351145 Ki > 100000 nM T79961 CV1U7L 73352414 Ki = 2996 nM T79961 C87LGB 73352415 Ki = 2417 nM T79961 C4F7VK 73355415 Ki = 595 nM T79961 CHV3W1 73774630 EC50 > 30000 nM T79961 C8IDL3 75306277 Ki = 794.33 nM T79961 C43NME 76313419 EC50 = 2800 nM T79961 C5JNZ1 76324306 EC50 = 4200 nM T79961 C2BM9L 89768534 EC50 > 30000 nM T79961 CB4Y7R 89768546 EC50 > 30000 nM T79961 CYX9R8 89777050 EC50 > 10000 nM T79961 C5MR9K 89777151 EC50 > 30000 nM T79961 CY1F7W 90510721 IC50 > 10000 nM T79961 C4RUP2 101882890 Ki = 2.951 nM T79961 CC3YS5 118706050 Ki > 100000 nM T79961 C6DXV9 118706052 Ki > 100000 nM T79961 CL4EO9 118706054 Ki = 41686.94 nM T79961 CG86QX 118710659 Ki = 87.1 nM T79961 C9D1MC 118710661 Ki = 16.6 nM T79961 C9H7FI 118710663 Ki = 19.5 nM T79961 CV2JU4 118710665 Ki = 20.89 nM T79961 C97VPM 118710667 Ki = 16.98 nM T79961 CI26PL 118710669 Ki = 5.495 nM T79961 C1OV8Y 118710671 Ki = 120.23 nM T79961 CBA78Q 118712533 EC50 > 10000 nM T79961 CQ5BG0 118712534 EC50 = 1800 nM T79961 C71SFO 118712535 EC50 = 150 nM T79961 CJ86QL 118712536 EC50 = 120 nM T79961 C49WAF 118712537 EC50 = 120 nM T79961 C0IFX1 118712538 EC50 = 128.82 nM T79961 C5LFW4 118717221 Ki > 1000 nM T79961 C67JND 118719476 IC50 > 30000 nM T79961 C43OWC 118719477 IC50 = 1300 nM T79961 C67AZQ 118719478 IC50 = 3300 nM T79961 C6GC1X 118719479 IC50 = 5500 nM T79961 CO48KZ 118719480 IC50 = 1200 nM T79961 C3S8YR 118719481 IC50 = 2700 nM T79961 C5DLN6 118719482 IC50 = 2000 nM T79961 C5F2GO 118719483 IC50 = 1300 nM T79961 CY3P9O 118719484 IC50 > 30000 nM T79961 C3O6SF 118719485 IC50 = 2400 nM T79961 CRJ80C 118719486 IC50 = 1000 nM T79961 C5J0ZO 118719487 IC50 > 30000 nM T79961 CGX78T 118719488 IC50 = 1400 nM T79961 C8B5EP 118719489 IC50 = 510 nM T79961 CWA8L6 118719490 IC50 = 700 nM T79961 CG8VZ1 118719491 IC50 = 1600 nM T79961 CWUO95 118719492 IC50 = 900 nM T79961 C8H6OP 118719493 IC50 = 4100 nM T79961 CU9K8V 118719494 IC50 = 1900 nM T79961 CWSM78 118719495 IC50 = 1100 nM T79961 C3HP2B 118719496 IC50 = 3200 nM T79961 C8OH4B 118719497 IC50 = 3300 nM T79961 CZ6T4H 118719498 IC50 = 1300 nM T79961 CD6K4Q 118719499 IC50 = 1300 nM T79961 CNG28F 118719500 IC50 = 6400 nM T79961 CCK73A 118719501 IC50 = 2200 nM T79961 C4JY5S 118719502 IC50 = 263.03 nM T79961 CI8CR0 118719920 Ki = 102.33 nM T79961 CV1WX5 118719921 Ki = 5.623 nM T79961 CIAG59 118719922 Ki = 2.291 nM T79961 CC5Q8Y 118719923 Ki = 8.71 nM T79961 CC8R6U 118719924 Ki = 30.9 nM T79961 CT8KO4 118719925 Ki = 14454.4 nM T79961 C16DHZ 118719926 Ki = 4570.88 nM T79961 CLA06I 118719927 Ki = 3090.3 nM T79961 CF20SR 118719928 Ki = 851.14 nM T79961 C6N7HV 118719929 Ki = 346.74 nM T79961 C64BIA 118719930 Ki = 338.84 nM T79961 CG4ZV5 118719931 Ki = 48.98 nM T79961 C05OBV 118723724 Ki > 100000 nM T79961 COA1Z8 118724894 IC50 > 10000 nM T79961 CB60YL 118724895 IC50 = 850 nM T79961 CJTN16 118724896 IC50 = 610 nM T79961 C2Y1MB 118724897 IC50 = 5888.44 nM T79961 CPH27Q 118724898 IC50 < 10000 nM T79961 CL47KT 118724899 IC50 < 10000 nM T79961 C6Z0AW 118724900 IC50 = 5623.41 nM T79961 C2WR3S 118724901 IC50 = 1600 nM T79961 C6NZO1 118724902 IC50 < 10000 nM T79961 C5YIG7 118724903 IC50 = 2100 nM T79961 CPZE10 118724904 IC50 = 2400 nM T79961 C6Z9LV 118724905 IC50 < 10000 nM T79961 CA0FH7 118724906 IC50 > 10000 nM T79961 CQ12NM 118724907 IC50 > 10000 nM T79961 CQ89TM 118724908 IC50 > 10000 nM T79961 C31FGS 118724909 IC50 < 10000 nM T79961 CQ5U0O 118724910 IC50 > 10000 nM T79961 CN15JW 118724911 IC50 = 3200 nM T79961 CX90IL 122194369 Ki = 6950 nM T79961 CU0B9P 122194370 Ki = 870 nM T79961 C79UOH 122194371 Ki > 30000 nM T79961 CMY91C 122194372 Ki = 6970 nM T79961 CCDI50 122194373 Ki = 2140 nM T79961 C3JI4Q 122194374 Ki = 380 nM T79961 CA6M5R 122194375 Ki > 10000 nM T79961 C7M1QH 122194376 Ki = 1810 nM T79961 C1JB0D 122194377 Ki = 5410 nM T79961 CD5NB9 122194378 Ki = 2050 nM T79961 C8O1QD 122194379 Ki > 10000 nM T79961 CFYZ56 122194380 Ki = 4300 nM T79961 C7ODW3 122195524 Ki > 900 nM T79961 C8MC1I 127028408 Ki = 2818.38 nM T79961 CJ2O5A 127044078 EC50 > 10000 nM T79961 CJ94GK 129316454 EC50 > 10000 nM T79961 CGHO19 132060770 Ki = 2591 nM T79961 CT81OY 132060776 Ki = 2471 nM T79961 CAVB41 132584404 Ki > 10000 nM T79961 CBU81N 134149168 Ki = 3493 nM T79961 CK64BF 134824563 IC50 = 1174.9 nM T79961 C4UX2M 135430667 Ki = 6165.95 nM T79961 CC3AT8 137631491 IC50 = 1445.44 nM T79961 CQ7JO0 137632697 IC50 = 6025.6 nM T79961 CW3M1T 137634701 IC50 = 8709.64 nM T79961 C6QB9W 137635734 Ki = 7943.28 nM T79961 CX8O0V 137636308 Ki = 9120.11 nM T79961 CH1G9Z 137636320 IC50 < 10000 nM T79961 C8KB2A 137636421 IC50 = 7762.47 nM T79961 CJ17IA 137637123 IC50 = 7244.36 nM T79961 C7VUW4 137637944 IC50 = 510 nM T79961 CY8Q1V 137638270 IC50 = 1030 nM T79961 C4VMA3 137638421 IC50 = 3388.44 nM T79961 CK6WQ5 137640100 IC50 = 1778.28 nM T79961 CZ4TA9 137640201 Ki = 3715.35 nM T79961 CX4A3N 137640511 Ki = 23988.33 nM T79961 CV7HT3 137641540 IC50 = 1445.44 nM T79961 C4Q6ZM 137642607 Ki = 2041.74 nM T79961 C4PU6H 137643771 IC50 = 4466.84 nM T79961 C0KL6Q 137644962 Ki = 6025.6 nM T79961 CTM03J 137645753 IC50 = 3019.95 nM T79961 CG8P6I 137645938 Ki = 3548.13 nM T79961 C2XMK6 137647734 IC50 = 695 nM T79961 C60FEV 137648229 IC50 = 4010 nM T79961 C1ZMO8 137648371 IC50 = 6760.83 nM T79961 C76ITZ 137650577 IC50 = 6309.57 nM T79961 CBN1K6 137650836 Ki = 77.62 nM T79961 CWG87E 137651507 Ki = 3800 nM T79961 C51PZY 137653721 IC50 = 1819.7 nM T79961 C61WAG 137654353 IC50 = 1130 nM T79961 CWOV78 137655063 IC50 = 732 nM T79961 CUC54G 137655636 Ki = 758.58 nM T79961 CB1C8A 137656435 IC50 = 4265.8 nM T79961 CEM27S 137658629 IC50 = 1288.25 nM T79961 CJ19YA 137660071 IC50 = 3467.37 nM T79961 CP7V9K 137661122 IC50 > 10000 nM T79961 C68QKL 137661317 Ki = 22.91 nM T79961 CDA8V2 137661377 Ki = 1949.84 nM T79961 C41ZYJ 137701968 EC50 > 30000 nM T79961 CXWJ63 139414008 EC50 = 1300 nM T79961 C38OTS 145960427 Ki = 467.74 nM T79961 C06LVP 145960466 Ki = 19.05 nM T79961 CSV5D4 145960592 Ki = 245.47 nM T79961 C4KH9G 145960827 Ki = 112.2 nM T79961 CJI6G2 145961125 Ki = 1949.84 nM T79961 CK7OJ5 145961126 Ki = 1288.25 nM T79961 C0XL7S 145961152 Ki = 10715.19 nM T79961 C3WFT9 145961161 Ki = 45.71 nM T79961 CJ50OV 145961495 Ki = 363.08 nM T79961 CAH97Y 145961981 Ki = 1096.48 nM T79961 CH1AE6 145962050 Ki = 1122.02 nM T79961 CG16NQ 145963288 Ki = 630.96 nM T79961 C6P3SR 153287553 Ki > 10000 nM T79961 CV9G7Z 153287572 Ki > 10000 nM T79961 CO85KL 153287574 Ki > 10000 nM T79961 CJKG35 155510347 Ki = 4490 nM T79961 C8IXK6 155511112 Ki = 640 nM T79961 CY83UA 155511167 Ki = 130 nM T79961 C2BDK6 155513985 Ki = 162.18 nM T79961 C08ASW 155515327 IC50 > 10000 nM T79961 C6JSC8 155515662 Ki = 150 nM T79961 CJG12Y 155516095 Ki = 470 nM T79961 C53FKW 155516382 Ki = 223.87 nM T79961 CI24NW 155516845 Ki = 260 nM T79961 C0JM8H 155518181 Ki = 60 nM T79961 C0MT4Q 155519740 Ki = 33.88 nM T79961 CUSA24 155519891 Ki > 10000 nM T79961 C4B7VK 155520267 Ki = 150 nM T79961 CPVA65 155521382 Ki = 977.24 nM T79961 C9N3JA 155521639 Ki = 1610 nM T79961 C7HPL3 155521847 Ki = 80 nM T79961 CFVP27 155521893 Ki = 141.25 nM T79961 CL9ET5 155522354 Ki = 426.58 nM T79961 CL6O1R 155523647 Ki = 38.9 nM T79961 C38PTA 155523888 Ki = 426.58 nM T79961 C8AMH9 155524478 Ki = 260 nM T79961 C6PFY7 155524809 Ki = 240 nM T79961 C5P1YE 155525064 Ki = 1348.96 nM T79961 CDQ89Y 155525097 Ki = 33.88 nM T79961 C7EIK1 155525691 Ki = 190 nM T79961 CBK0Y7 155528269 Ki = 501.19 nM T79961 CPG08Y 155528419 Ki = 230 nM T79961 CRPY78 155529196 Ki = 30 nM T79961 CUT8S5 155530448 IC50 > 10000 nM T79961 C7CU8J 155535606 Ki = 109.65 nM T79961 CK91NV 155535972 Ki = 60 nM T79961 CB79ZW 155536080 Ki > 10000 nM T79961 C2XN8P 155536739 Ki = 40 nM T79961 CV2NG9 155539712 Ki = 29.51 nM T79961 CY2L3J 155540315 Ki = 380 nM T79961 CY4SX1 155541234 IC50 > 10000 nM T79961 CK70MJ 155541812 Ki = 1.8 nM T79961 CF50KG 155542317 IC50 > 10000 nM T79961 CS5YB1 155543344 Ki = 208.93 nM T79961 COV93Z 155543943 Ki = 239.88 nM T79961 CX4J2Q 155545295 IC50 > 10000 nM T79961 C2CB8H 155548585 Ki = 2398.83 nM T79961 C1XIA4 155549890 Ki = 1050 nM T79961 C9KBH7 155550435 Ki = 70.79 nM T79961 CRIJ70 155550631 Ki = 112.2 nM T79961 CR8XF7 155551306 Ki = 130 nM T79961 CW92JZ 155551421 Ki = 1370 nM T79961 COF49W 155551902 Ki = 7079.46 nM T79961 CXZQ46 155552922 Ki = 707.95 nM T79961 CE70NU 155553089 Ki = 240 nM T79961 CS1DK6 155554149 Ki = 40 nM T79961 C7TF1D 155554261 Ki = 58.88 nM T79961 C73DFN 155554567 Ki = 457.09 nM T79961 C1TDY8 155556289 Ki = 95.5 nM T79961 C2D3SP 155557118 Ki = 120.23 nM T79961 C75PXS 155559290 Ki = 1513.56 nM T79961 CEAD84 155559740 Ki = 74.13 nM T79961 CP2U8A 155560012 Ki = 199.53 nM T79961 CU3TF1 155560139 Ki = 363.08 nM T79961 CCO15D 155560304 Ki = 295.12 nM T79961 CMX98Q 155562285 Ki = 10 nM T79961 C7P2OG 155562295 Ki = 550 nM T79961 CDYV69 155562882 Ki = 260 nM T79961 C8WE2F 155563061 Ki = 3490 nM T79961 C2G7UH 155565074 Ki = 100 nM T79961 CVLR58 155565285 Ki = 1202.26 nM T79961 C9AF7I 155565770 Ki = 65 nM T79961 CDS7K2 155566289 Ki = 295.12 nM T79961 CY30EN 155567379 Ki = 30.9 nM T79961 C3N9VU 10251906 Ki > 500 nM T79961 C9RLJ3 3661 Ki = 0.6 nM T79961 CD6OK3 44455198 Ki = 17.5 nM T79961 D02BOW 5926 Ki = 3801.89 nM T79961 D02EXX 3013846 Ki = 1180 nM T79961 D02KZD 71598521 IC50 = 300 nM T79961 D02ZPV 10125445 Ki = 63.1 nM T79961 D03DKZ 42633508 Ki = 159 nM T79961 D05ZUX 44207909 Ki >= 1000 nM T79961 D06IUC 6508730 Ki = 228 nM T79961 D07GPQ 132947 Ki = 33.88 nM T79961 D09RPR 16737207 Ki > 10000 nM T79961 D0A2KT 3014059 Ki = 0.22 nM T79961 D0AR0H 6508724 Ki = 83 nM T79961 D0F5LH 4634 Ki = 14.13 nM T79961 D0F9QY 6604893 EC50 = 2600 nM T79961 D0FF6S 16038374 IC50 > 10000 nM T79961 D0G4CG 4629 EC50 = 2300 nM T79961 D0H8XV 12963076 Ki = 2691.53 nM T79961 D0HP1O 119357 Ki = 537.03 nM T79961 D0I9LU 2229 Ki = 933.25 nM T79961 D0JV2S 3008304 EC50 = 4080 nM T79961 D0L1XR 4630 EC50 = 55 nM T79961 D0N2KU 44517677 Ki = 1800 nM T79961 D0T2RY 9948320 Ki >= 1000 nM T79961 D0WO3A 4141 Ki = 6918.31 nM T79961 D0X7HD 11184481 Ki = 5200 nM T79961 D0Z5RQ 656392 IC50 = 1220 nM T79961 D0Z6VT 71737672 EC50 = 190 nM T00140 D02HWP 2722 IC50 = 3600 nM T00140 D03RTS 2662 IC50 > 10000 nM T00140 D04AIT 5280445 IC50 = 1600 nM T00140 D05VLS 5090 IC50 > 10000 nM T00140 D09JUG 60490 IC50 = 150 nM T00140 D0K8KX 5280343 IC50 = 790 nM T00140 D0MM8N 3686 IC50 > 10000 nM T00140 D0R1QE 3672 IC50 = 17000 nM T00140 D0R1RS 3715 IC50 = 7000 nM T00140 D0U5CE 1548943 IC50 = 56000 nM T00140 D0YG7M 3827 IC50 > 100000 nM T00140 D02WFN 46207733 IC50 = 4400 nM T00140 D04WMR 59757 EC50 = 70 nM T00140 D07SDQ 969516 IC50 = 30000 nM T00140 D08PXR 3086671 IC50 = 160 nM T00140 D0H7PW 638024 IC50 = 54000 nM T00140 D0U3EP 445154 IC50 = 4900 nM T00140 D0DK4I 4534 IC50 = 25 nM T00140 D0O4QB 3314 IC50 = 26000 nM T00140 D01DAD 9821945 IC50 = 230 nM T00140 D04TCU 9905233 IC50 = 117 nM T00140 D05HSW 3218 IC50 = 3500 nM T00140 D05MCS 44473151 IC50 = 20000 nM T00140 D05WPQ 6438354 IC50 = 13 nM T00140 D07HBI 132306 IC50 = 20 nM T00140 D09BKE 4553 IC50 > 10000 nM T00140 D0D8MD 132998 IC50 = 60 nM T00140 D0F8DL 176155 IC50 = 80 nM T00140 D0H7GH 131627 IC50 = 20 nM T00140 D0HJ1Y 5353454 IC50 = 80 nM T00140 D0IL8R 101018054 IC50 = 170 nM T00140 D0JY4Y 443292 IC50 = 100 nM T00140 D0K2ER 3651377 IC50 = 60 nM T00140 D0L1IH 178577 IC50 = 80 nM T00140 D0M0QX 23672584 IC50 = 8 nM T00140 D0N1SU 133021 IC50 = 180 nM T00140 D0O8ZE 5059 IC50 = 300 nM T00140 D0P3KA 60542 IC50 = 3000 nM T00140 D0QE5B 6436051 IC50 = 4860 nM T00140 D0S6VB 123723 IC50 = 60 nM T00140 D0S8YL 3969 IC50 = 18900 nM T00140 D0X9KE 71460 IC50 = 80 nM T00140 C85KQB 2202 IC50 = 7000 nM T00140 CQ0D8J 3469 IC50 = 75000 nM T00140 CZ9Y8R 8247 IC50 = 65000 nM T00140 CV24FH 10228 IC50 = 36200 nM T00140 C49FZU 11617 IC50 = 83000 nM T00140 CK6VT0 60923 IC50 = 1.6 nM T00140 CME3K9 65048 IC50 = 30400 nM T00140 CZ6F7S 67278 IC50 = 20 nM T00140 C0TY5F 72059 IC50 = 100 nM T00140 CKB4R0 73145 IC50 > 40000 nM T00140 CKH0W1 73170 IC50 > 40000 nM T00140 CQD56Z 73299 IC50 > 40000 nM T00140 CQT19P 73641 IC50 = 42000 nM T00140 CCJ6E2 75294 IC50 = 9400 nM T00140 CU4S9Z 80074 IC50 = 170 nM T00140 CUAW60 82755 IC50 = 13000 nM T00140 CV0Q6U 88281 IC50 = 2900 nM T00140 C5Z1QA 96028 IC50 > 200000 nM T00140 C94WZM 100659 IC50 = 2500 nM T00140 CHF2E5 101761 IC50 > 40000 nM T00140 CFT49L 122805 IC50 > 5000 nM T00140 CC8QV4 124072 IC50 = 3200 nM T00140 C3E0RZ 127576 IC50 = 25 nM T00140 C2D1AN 127577 IC50 = 90 nM T00140 CUP4Y3 128132 IC50 = 11 nM T00140 CPVH47 129065 IC50 = 230 nM T00140 C35GTR 129232 IC50 = 300 nM T00140 CK3V8F 130007 IC50 = 2100 nM T00140 CBG9Z6 131453 IC50 = 500 nM T00140 C42HZM 145696 IC50 = 230 nM T00140 CS74HZ 145726 IC50 = 1700 nM T00140 C1H8NR 155248 IC50 = 2350 nM T00140 C5GFP0 155948 IC50 > 200000 nM T00140 C83FUH 159969 IC50 = 2700 nM T00140 CV87RA 167846 IC50 = 770 nM T00140 CW8K1N 168928 IC50 > 40000 nM T00140 C7PU2J 171489 IC50 = 680 nM T00140 C7H1QR 182364 IC50 = 9300 nM T00140 CD3NR8 188382 IC50 = 6000 nM T00140 C13WSH 195771 IC50 = 45 nM T00140 C3YD0N 258337 IC50 = 500 nM T00140 CS4HK9 295563 IC50 = 4500 nM T00140 CB7GM0 323821 IC50 = 5100 nM T00140 C52UFN 345753 IC50 = 1800 nM T00140 C9CFX8 363127 IC50 = 250 nM T00140 CXV7H2 363128 IC50 = 70 nM T00140 C8Y9JE 363130 IC50 = 660 nM T00140 CD43EV 367858 IC50 = 700 nM T00140 C08BKG 392401 IC50 = 200 nM T00140 C0GPV1 402434 IC50 = 5300 nM T00140 C5CSG4 402435 IC50 = 4500 nM T00140 CUW26R 423227 IC50 = 2900 nM T00140 C8P3CK 427265 IC50 = 1900 nM T00140 CLR79X 442911 IC50 = 9300 nM T00140 C8AZ6K 460888 IC50 = 760 nM T00140 CMT3P0 480764 IC50 > 10000 nM T00140 CDCQ38 607148 IC50 > 50000 nM T00140 C27XBF 610243 IC50 = 1870 nM T00140 CA9BW2 637234 IC50 = 42000 nM T00140 CQ94TR 639465 IC50 = 50 nM T00140 CQ59SY 639665 IC50 = 2100 nM T00140 CQAV61 642530 IC50 = 200 nM T00140 CV97HM 663693 IC50 > 15000 nM T00140 CZ4O7G 664510 IC50 > 50000 nM T00140 CCYE09 675655 IC50 = 24600 nM T00140 CS43TM 689163 IC50 = 2700 nM T00140 CW7J6K 697279 IC50 = 8300 nM T00140 CHXJ51 697280 IC50 = 300 nM T00140 C0WIK8 697307 IC50 = 15300 nM T00140 C86DSV 698943 IC50 = 400 nM T00140 C8U2TS 702098 IC50 > 30000 nM T00140 CF1I2C 715201 IC50 = 7600 nM T00140 CDCF89 715217 IC50 = 20000 nM T00140 C9O6KL 717261 IC50 = 480 nM T00140 CF9J2K 717265 IC50 = 300 nM T00140 CRTJ63 717270 IC50 = 3000 nM T00140 C1S4ER 744225 IC50 = 66000 nM T00140 CG0JL1 747904 IC50 = 2200 nM T00140 CJ8A2B 767605 IC50 = 730 nM T00140 C0SBW6 768022 IC50 = 400 nM T00140 CPM12N 775994 IC50 > 100000 nM T00140 CB59GS 778729 IC50 = 8200 nM T00140 CODL04 788760 IC50 = 2000 nM T00140 C1PD4J 805589 IC50 = 8100 nM T00140 CL4AH7 809033 IC50 = 600 nM T00140 C48FJV 809037 IC50 = 1300 nM T00140 CNYT14 809076 IC50 = 430 nM T00140 C7Q4HC 814008 IC50 = 4600 nM T00140 C6YN0T 856589 IC50 = 1800 nM T00140 CC9MG8 856590 IC50 = 600 nM T00140 CR0UW1 856592 IC50 = 2100 nM T00140 C4Z9YR 856602 IC50 = 900 nM T00140 C0J3IM 861855 IC50 = 16000 nM T00140 CQ7A4Z 871145 IC50 = 3300 nM T00140 C4MT1H 871502 IC50 = 237000 nM T00140 C7U3CX 873133 IC50 = 50 nM T00140 C6G8QZ 877802 IC50 = 1200 nM T00140 CHX2D5 877815 IC50 = 30 nM T00140 CVB9K6 882228 IC50 = 2400 nM T00140 C8FH0Q 886842 IC50 = 1400 nM T00140 CFP6W9 887113 IC50 = 60 nM T00140 C09JDB 924716 IC50 = 36000 nM T00140 CR3FK1 932731 IC50 = 3800 nM T00140 CLCG81 938024 IC50 = 7000 nM T00140 CZB2G9 972713 IC50 = 600 nM T00140 C9AXN3 972868 IC50 = 60 nM T00140 CQX7D3 980457 IC50 = 160 nM T00140 C1I9LG 987980 IC50 = 29000 nM T00140 C2G8DI 993074 IC50 = 44000 nM T00140 CEJ25S 996799 IC50 = 45000 nM T00140 CECO79 1017552 IC50 = 15000 nM T00140 CE4HM8 1032885 IC50 = 850 nM T00140 C3TGX9 1040851 IC50 = 2800 nM T00140 C0SGD7 1071670 IC50 = 7700 nM T00140 CP8ZQ5 1079369 IC50 = 420 nM T00140 CA1TU5 1079729 IC50 > 200000 nM T00140 CP8ZL1 1094081 IC50 = 2300 nM T00140 CFOD51 1115445 IC50 = 48000 nM T00140 CP8RV2 1154253 IC50 = 80 nM T00140 CVD4F7 1154287 IC50 = 900 nM T00140 CQ1PV5 1205608 IC50 > 5000 nM T00140 CLKQ75 1206916 IC50 = 470 nM T00140 CE3AH6 1219517 IC50 = 20000 nM T00140 CR0U5L 1220478 IC50 = 89000 nM T00140 C90XUW 1221901 IC50 = 1250 nM T00140 C5H0SF 1225140 IC50 = 300 nM T00140 C52EOR 1229519 IC50 = 68000 nM T00140 C4APY7 1237983 IC50 = 67000 nM T00140 CWA0B4 1240120 IC50 = 4700 nM T00140 CCS7L3 1309076 IC50 = 76000 nM T00140 CILN42 1356792 IC50 > 10000 nM T00140 CGBU23 1433361 IC50 = 1800 nM T00140 CEHU17 1442508 IC50 = 400 nM T00140 C1RD3X 1548457 IC50 = 1100 nM T00140 C6HL7N 1639245 IC50 > 30000 nM T00140 CS8UR4 1718584 IC50 = 980 nM T00140 CFE92U 1723288 IC50 = 800 nM T00140 C72GZQ 1732961 IC50 = 80000 nM T00140 CQJ19K 1733195 IC50 = 14200 nM T00140 CUS89M 1733918 IC50 = 14000 nM T00140 C16VCG 1742972 IC50 = 2700 nM T00140 C1DKO0 1749337 IC50 = 2450 nM T00140 CYFZ69 1811377 IC50 = 800 nM T00140 C9Q6RD 1816908 IC50 = 37500 nM T00140 CM3X2R 1822643 IC50 = 1040 nM T00140 C1V6AQ 1823617 IC50 = 33800 nM T00140 C3NR4Z 1913485 IC50 = 3500 nM T00140 CC25XB 1998811 IC50 > 20000 nM T00140 CNPK95 2215254 IC50 = 4900 nM T00140 CTK8A2 2246826 IC50 = 860 nM T00140 CJGB03 2249763 IC50 = 900 nM T00140 C8ME9W 2253173 IC50 = 160 nM T00140 C2WFK8 2281220 IC50 = 300 nM T00140 CKG9S3 2354998 IC50 = 2300 nM T00140 CZ2X9Q 2718951 IC50 = 230 nM T00140 C2VP6M 2750392 IC50 = 52000 nM T00140 C8E1MI 2801550 IC50 = 1100 nM T00140 C9RFE2 2806778 IC50 = 700 nM T00140 C45LQX 2841002 IC50 = 12300 nM T00140 CDQ97L 2883254 IC50 > 50000 nM T00140 C60OPF 2883266 IC50 = 240 nM T00140 CD0X5M 2920571 IC50 > 100000 nM T00140 CU16KY 2920793 IC50 > 100000 nM T00140 CL1QK7 2962247 IC50 = 65000 nM T00140 C9S5KI 2971957 IC50 = 97000 nM T00140 CQM64G 3037018 IC50 = 2800 nM T00140 CG0MN3 3080635 IC50 = 25100 nM T00140 CUY83X 3094561 IC50 = 34 nM T00140 CVU5O1 3108985 IC50 = 2800 nM T00140 CY2Z6S 3116544 IC50 = 4 nM T00140 C1OTU9 3136123 IC50 > 100000 nM T00140 C3G9QL 3136134 IC50 > 100000 nM T00140 CQSX43 3136217 IC50 = 81000 nM T00140 CSQN24 3159469 IC50 = 2700 nM T00140 C1WVJ3 3385224 IC50 = 8000 nM T00140 CNOE15 3667020 IC50 = 1000 nM T00140 CHZ9Q0 3684695 IC50 = 8000 nM T00140 C2H7AN 3684697 IC50 = 2000 nM T00140 CRL9T0 3684699 IC50 = 3000 nM T00140 C3KUC1 3684700 IC50 = 600 nM T00140 CO9A3L 3692652 IC50 = 6000 nM T00140 CZ7K1O 3735492 IC50 = 1000 nM T00140 CKQ06A 3765426 IC50 = 5000 nM T00140 CZP0H9 3775015 IC50 = 3700 nM T00140 CRV1K2 3861394 IC50 = 800 nM T00140 CYI61N 4078425 IC50 = 33 nM T00140 CT4BD9 4143121 IC50 = 1700 nM T00140 CRFA96 4149421 IC50 = 500 nM T00140 C4W9DQ 4187769 IC50 = 230 nM T00140 CE18AL 4196858 IC50 = 11000 nM T00140 C2DN4A 4228320 IC50 > 50000 nM T00140 CF4G5U 4443437 IC50 = 3000 nM T00140 CJ9T7B 4517796 IC50 = 1300 nM T00140 C5B4DK 4519262 IC50 = 1100 nM T00140 CGP1T5 4556427 IC50 = 610 nM T00140 CZ9E1B 4560409 IC50 = 230 nM T00140 CJ0D1G 4589007 IC50 = 8000 nM T00140 C4E3MH 4645817 IC50 = 8600 nM T00140 C2X3FK 4665555 IC50 = 4000 nM T00140 CK98IS 4690153 IC50 > 50000 nM T00140 C50WLT 4968501 IC50 = 3100 nM T00140 CC4T0L 4984206 IC50 = 70000 nM T00140 C3XJI9 4984595 IC50 = 270 nM T00140 CIH29P 5036963 IC50 = 10 nM T00140 C1ON0D 5061725 IC50 = 5500 nM T00140 C9C8GI 5061930 IC50 = 53000 nM T00140 C6PB0T 5086864 IC50 = 590 nM T00140 CXT8B4 5104845 IC50 = 1300 nM T00140 C6H2SP 5185168 IC50 = 9800 nM T00140 CF3NM8 5280701 IC50 > 100000 nM T00140 C0D3PO 5281671 IC50 = 100000 nM T00140 CZM7D8 5281794 IC50 = 7400 nM T00140 CKER75 5283133 EC50 = 3 nM T00140 C2NKF5 5283162 IC50 > 50000 nM T00140 C34ZQB 5318477 IC50 = 1000 nM T00140 CC3QF0 5321018 IC50 > 200000 nM T00140 C2J3TK 5335462 IC50 = 1130 nM T00140 C17NYJ 5350310 IC50 = 3000 nM T00140 C84IDS 5373044 IC50 > 30000 nM T00140 CFEC26 5374732 IC50 > 10000 nM T00140 CLA6Y8 5411248 IC50 = 300 nM T00140 CL52GB 5411269 IC50 > 30000 nM T00140 CID17E 5455586 IC50 = 350 nM T00140 COR5X4 5466621 IC50 = 4100 nM T00140 CQB12M 5757474 IC50 = 130 nM T00140 C9LYS8 5760413 IC50 = 800 nM T00140 C3IP5M 5809575 IC50 = 70 nM T00140 C5M0AJ 5909099 IC50 = 330 nM T00140 C2TU6H 5983898 IC50 = 530 nM T00140 CXL1P5 5997630 IC50 = 6100 nM T00140 CC3V5A 6229062 IC50 = 17000 nM T00140 C0BY6F 6261723 IC50 > 50000 nM T00140 C3G7DT 6365297 IC50 = 100 nM T00140 C40FZG 6366698 IC50 = 240 nM T00140 C02AQY 6366699 IC50 < 1000 nM T00140 C3KY7T 6375919 IC50 = 30000 nM T00140 CWK1F9 6438990 IC50 = 690 nM T00140 C62UOZ 6439221 IC50 = 54 nM T00140 CHQ4Z3 6439222 IC50 = 120 nM T00140 COC86Q 6439421 IC50 = 770 nM T00140 CLJ91K 6439912 IC50 = 1700 nM T00140 CQO9T1 6440631 IC50 > 50000 nM T00140 CQZ8U3 6446027 IC50 > 100000 nM T00140 CXZC29 6610350 IC50 = 200 nM T00140 C9A0PS 6871421 IC50 = 620 nM T00140 CI8Y4V 6874154 IC50 = 5400 nM T00140 CQ31FO 7034541 IC50 = 1100 nM T00140 CB8JA2 7038010 IC50 > 50000 nM T00140 C6FH9C 7299191 IC50 = 1800 nM T00140 C9EY3W 7341803 IC50 = 500 nM T00140 C82TEX 7515046 IC50 > 1000 nM T00140 CYOI76 8765451 IC50 = 1600 nM T00140 CGA06D 9507010 IC50 = 70000 nM T00140 CA57OF 9796542 IC50 = 160 nM T00140 C9WR3H 9797751 IC50 = 85 nM T00140 C3HYJ6 9799029 IC50 = 930 nM T00140 CV8G7C 9803626 IC50 900 nM T00140 CA7MG6 9803993 IC50 = 20 nM T00140 CMPU43 9805176 IC50 = 14 nM T00140 CUS6L8 9822795 IC50 = 110 nM T00140 CQ1IV3 9831104 IC50 = 18 nM T00140 C6GSZ2 9836535 IC50 = 300 nM T00140 C83VNA 9841863 IC50 = 580 nM T00140 CKG7X0 9847369 IC50 = 115 nM T00140 C6VD1C 9847616 IC50 = 27 nM T00140 CON54H 9848282 IC50 = 526 nM T00140 C28IUE 9850828 IC50 = 89 nM T00140 CS6Y5U 9861661 IC50 = 8000 nM T00140 C2Y4XH 9867465 IC50 = 15 nM T00140 CJIF86 9867467 IC50 = 8 nM T00140 CF7M2Y 9870460 IC50 = 310 nM T00140 C2TUG6 9872445 IC50 = 185 nM T00140 CE3S8I 9874478 IC50 = 26 nM T00140 C7RVN8 9883481 IC50 = 200 nM T00140 C3RJ8S 9884093 IC50 = 100 nM T00140 CTF3X0 9885237 IC50 = 3400 nM T00140 CRH61A 9890796 IC50 = 70 nM T00140 CZ3SA4 9891815 IC50 = 7 nM T00140 CS7HU2 9902041 IC50 = 50 nM T00140 CT82WH 9904992 IC50 = 170 nM T00140 C0RO9L 9905075 IC50 = 200 nM T00140 CRU80N 9910119 IC50 = 89 nM T00140 CNI49H 9913604 IC50 = 420 nM T00140 CKD2U1 9914988 IC50 = 358 nM T00140 CQAU05 9917207 IC50 = 8 nM T00140 CHD5A1 9921059 IC50 = 3200 nM T00140 COTJ38 9926352 IC50 = 190 nM T00140 CZSF75 9926487 IC50 = 50 nM T00140 CI5Y3Z 9929628 IC50 = 40 nM T00140 C36SEC 9931329 IC50 = 340 nM T00140 CKWB53 9947925 IC50 > 50000 nM T00140 C2PAC8 9958732 IC50 = 213 nM T00140 CX98TO 9968732 IC50 = 350 nM T00140 C3W4LQ 9969506 IC50 = 80 nM T00140 C2TO9Y 9977187 IC50 = 330 nM T00140 CJ5FC4 9977253 IC50 = 1100 nM T00140 CV2X7O 9978273 IC50 = 70 nM T00140 CAMY05 9979136 IC50 = 210 nM T00140 CWK52R 9982617 IC50 = 20 nM T00140 CL86GV 9986780 IC50 = 900 nM T00140 CI3M8G 9995876 IC50 = 120 nM T00140 C9R8SY 10001795 IC50 = 160 nM T00140 CHFC56 10009283 IC50 = 60 nM T00140 CU7M8Q 10022483 IC50 = 150 nM T00140 C6HD9T 10022493 IC50 = 270 nM T00140 C6G2CK 10022494 IC50 = 150 nM T00140 CS6N7G 10024069 IC50 = 10 nM T00140 C2TS7E 10026136 IC50 = 410 nM T00140 C1N3OT 10029694 IC50 = 160 nM T00140 C6Y4ZJ 10031902 IC50 = 50 nM T00140 CDTE34 10038868 IC50 = 50 nM T00140 CCA7O1 10046101 IC50 = 170 nM T00140 C03EXZ 10046767 IC50 = 30 nM T00140 CL98OS 10051425 IC50 = 170 nM T00140 CK38OV 10053402 IC50 = 37 nM T00140 C6R7ZM 10054908 IC50 = 300 nM T00140 CD6J5Y 10059051 IC50 = 4800 nM T00140 CU3JK1 10065203 IC50 = 480 nM T00140 CVFI72 10069970 IC50 = 740 nM T00140 C86JOY 10070092 IC50 = 1900 nM T00140 C9GX7L 10070723 IC50 = 3220 nM T00140 CUZ91W 10071605 IC50 = 50 nM T00140 CVO16U 10071652 IC50 = 120 nM T00140 C8TEO4 10071695 IC50 = 1300 nM T00140 CQ9K7Y 10087103 IC50 = 390 nM T00140 CKBF18 10090114 IC50 = 440 nM T00140 CMY02E 10091294 IC50 = 220 nM T00140 C7QJL6 10100308 IC50 = 105 nM T00140 CH45QJ 10126163 IC50 = 820 nM T00140 CT7O8H 10130205 IC50 = 5800 nM T00140 CY6E8O 10133915 IC50 = 370 nM T00140 C1YCK6 10134800 IC50 = 1000 nM T00140 CDWT62 10172850 IC50 = 650 nM T00140 CS7N3M 10194182 IC50 = 620 nM T00140 CO7S9H 10200992 IC50 = 80 nM T00140 CGAP51 10215420 IC50 = 400 nM T00140 CQ5A1X 10219499 IC50 = 900 nM T00140 CBL7R3 10220019 IC50 = 1200 nM T00140 C67DXM 10220327 IC50 = 500 nM T00140 C14SLX 10242717 IC50 = 15000 nM T00140 CU8G6W 10244247 IC50 = 600 nM T00140 C8MFT2 10247254 IC50 = 390 nM T00140 C7H8QV 10249130 IC50 = 2300 nM T00140 C9CQ5K 10250327 IC50 = 520 nM T00140 CJT2W8 10258201 IC50 = 4000 nM T00140 C26GNO 10259199 IC50 = 20 nM T00140 CLZG02 10273406 IC50 = 290 nM T00140 CMAI02 10287180 IC50 = 700 nM T00140 C7TN1U 10287181 IC50 = 710 nM T00140 CXNL69 10287409 IC50 = 740 nM T00140 C5PYF7 10309829 IC50 = 650 nM T00140 C4J9ON 10309830 IC50 = 770 nM T00140 CWLK92 10314553 IC50 = 98 nM T00140 CR8ZA4 10317471 IC50 = 1180 nM T00140 CX4E1F 10326828 IC50 = 120 nM T00140 C1LZ7Y 10335263 IC50 = 50000 nM T00140 CP3AO1 10337829 IC50 = 600 nM T00140 CU82ZD 10338075 IC50 > 10000 nM T00140 C61ZNX 10341647 IC50 = 110 nM T00140 CPR1B0 10343085 IC50 = 4500 nM T00140 CN05LT 10344369 IC50 = 640 nM T00140 C63RGN 10347051 IC50 = 48 nM T00140 CK72OY 10348803 IC50 = 20 nM T00140 CJ4ZO7 10355545 IC50 > 50000 nM T00140 CKV03T 10356315 IC50 = 1200 nM T00140 CSGD92 10358121 IC50 = 3500 nM T00140 C8UN0D 10362302 IC50 = 6210 nM T00140 CSQJ68 10362915 IC50 = 1300 nM T00140 CP8HJ9 10375026 IC50 = 2700 nM T00140 CA8KG1 10380906 IC50 = 2700 nM T00140 C9CJY4 10381501 IC50 = 8000 nM T00140 CXB7N9 10385788 IC50 = 100 nM T00140 C47QCI 10386055 IC50 = 60 nM T00140 C4A8GJ 10391979 IC50 = 50 nM T00140 C4LJU3 10393783 IC50 = 250 nM T00140 C68HWP 10394023 IC50 = 55 nM T00140 CBOE34 10400378 IC50 = 1600 nM T00140 CGR03F 10404623 IC50 = 170 nM T00140 CK5A8R 10409943 IC50 = 70 nM T00140 CUFQ24 10422904 IC50 = 5000 nM T00140 CG8L4R 10427847 IC50 = 1000 nM T00140 CX5R2U 10429672 IC50 = 9900 nM T00140 CBI2R4 10429760 IC50 = 70 nM T00140 CFS98Y 10431646 IC50 = 840 nM T00140 CR08WG 10438989 IC50 = 70 nM T00140 CE3H4I 10443576 IC50 = 2200 nM T00140 C6TEG8 10450182 IC50 = 50 nM T00140 C31WQZ 10453108 IC50 = 60 nM T00140 C63NSV 10454188 IC50 = 60 nM T00140 CV3EP5 10454404 IC50 = 340 nM T00140 C1WM2V 10459826 IC50 = 3 nM T00140 C8V5TL 10461840 IC50 = 40 nM T00140 C02BUX 10475519 IC50 = 2800 nM T00140 CCWM91 10480128 IC50 = 1510 nM T00140 CEQ4U9 10484776 IC50 = 22 nM T00140 C6QRC5 10487728 IC50 = 940 nM T00140 CT8JS0 10487791 IC50 = 2400 nM T00140 CD06BK 10492504 IC50 = 5500 nM T00140 CLP06F 10493616 IC50 = 12000 nM T00140 COH23F 10495686 IC50 = 5000 nM T00140 C64YJH 10500489 IC50 = 380 nM T00140 C8N0BC 10501407 IC50 = 30 nM T00140 CN5Z2A 10502126 IC50 = 17 nM T00140 CT1X6K 10502533 IC50 = 70 nM T00140 CZS4N6 10503542 IC50 = 50 nM T00140 C8X7GV 10503635 IC50 = 20 nM T00140 CJU97M 10504173 IC50 = 17 nM T00140 C6YNZ3 10504174 IC50 = 20 nM T00140 CUG6X8 10504337 IC50 = 20 nM T00140 CV42CK 10504648 IC50 = 28 nM T00140 CHZ95J 10504790 IC50 = 14 nM T00140 CCM8L6 10505985 IC50 = 1065 nM T00140 C4R1GL 10507589 IC50 = 55 nM T00140 CGH9T4 10511759 IC50 = 1100 nM T00140 C3H8RS 10512076 IC50 = 1200 nM T00140 CBR68N 10513083 IC50 = 20000 nM T00140 CK63BA 10513218 IC50 = 7100 nM T00140 C5RZ8C 10513430 IC50 = 200 nM T00140 C6L7ZB 10514629 IC50 = 3400 nM T00140 CI6F7S 10516483 IC50 = 8500 nM T00140 CCO02A 10517413 IC50 > 50000 nM T00140 CCM82G 10525275 IC50 = 160 nM T00140 C23NYE 10525855 IC50 = 91 nM T00140 CTF1I2 10526411 IC50 = 27 nM T00140 CHYA29 10526644 IC50 = 820 nM T00140 CQDB43 10527066 IC50 = 30 nM T00140 CQSB28 10527551 IC50 = 20 nM T00140 CT0M8L 10528876 IC50 = 20 nM T00140 C74IOH 10528894 IC50 = 490 nM T00140 C3R9HM 10529019 IC50 = 33 nM T00140 CMKG89 10529020 IC50 = 40 nM T00140 CFM40N 10529179 IC50 = 35 nM T00140 C4QCJ1 10534946 IC50 = 700 nM T00140 C8S1EQ 10535951 IC50 = 1800 nM T00140 CSN38I 10538130 IC50 = 1200 nM T00140 C9V2XW 10539265 IC50 = 37000 nM T00140 C54DWE 10541466 IC50 = 22000 nM T00140 C1I9ZN 10542532 IC50 = 70 nM T00140 CN6M2J 10543472 IC50 = 15000 nM T00140 C09HCY 10550678 IC50 = 33 nM T00140 CY3MB9 10550685 IC50 = 47 nM T00140 C2T8WB 10551361 IC50 = 20 nM T00140 C01XGU 10553682 IC50 = 35 nM T00140 CR5S3Y 10554606 IC50 = 90 nM T00140 C89BIT 10556454 IC50 = 30 nM T00140 CUL5Y6 10559707 IC50 = 2000 nM T00140 CKCA29 10559708 IC50 = 900 nM T00140 CT4Y9Z 10561299 IC50 = 3700 nM T00140 CUZ53C 10563147 IC50 = 120 nM T00140 C03JWM 10563230 IC50 = 8800 nM T00140 CR8F6S 10563513 IC50 = 4000 nM T00140 C0ZIN1 10574353 IC50 = 60 nM T00140 C6Y0NH 10574430 IC50 = 350 nM T00140 C32TXJ 10576488 IC50 = 59 nM T00140 C7BK6X 10576564 IC50 = 1000 nM T00140 CCU95E 10577992 IC50 = 43 nM T00140 C49IZG 10587216 IC50 = 4600 nM T00140 CH4IC1 10588079 IC50 = 5200 nM T00140 CT25IR 10591982 IC50 = 60 nM T00140 C2EI7V 10598005 IC50 = 290 nM T00140 C0D2KL 10598842 IC50 = 160 nM T00140 CB93YD 10600308 IC50 = 27 nM T00140 CG60MZ 10600373 IC50 = 10 nM T00140 C1G2ZC 10600523 IC50 = 351 nM T00140 C5LUS1 10601569 IC50 = 22 nM T00140 CL4B7I 10601732 IC50 = 181 nM T00140 C91XFQ 10604402 IC50 = 60 nM T00140 CJ8HW1 10604538 IC50 = 40 nM T00140 C4Y0OU 10607231 IC50 = 2100 nM T00140 CF1QU8 10607535 IC50 = 480 nM T00140 CD1T5O 10608019 IC50 = 550 nM T00140 CR40MH 10608595 IC50 = 850 nM T00140 CJQ3V9 10613437 IC50 = 60 nM T00140 CKF79C 10616899 IC50 = 110 nM T00140 CGP2K9 10620314 IC50 = 1200 nM T00140 C0LV4T 10623059 IC50 = 87 nM T00140 CJHA39 10623784 IC50 = 28 nM T00140 CQ2H9M 10625017 IC50 = 31 nM T00140 CNQ81U 10630626 IC50 = 1700 nM T00140 CYW0R6 10630975 IC50 = 1950 nM T00140 C3U8NO 10632239 IC50 = 6000 nM T00140 C8KH9T 10633035 IC50 = 1600 nM T00140 CQ0A1J 10634989 IC50 = 420 nM T00140 CAO27K 10635787 IC50 = 3700 nM T00140 C72VDH 10636949 IC50 = 360 nM T00140 CXTZ76 10637675 IC50 = 160 nM T00140 C5N1ZT 10637982 IC50 = 30000 nM T00140 CL6T2N 10638828 IC50 = 20900 nM T00140 CA0KO6 10644762 IC50 = 6100 nM T00140 CWE21L 10645701 IC50 = 16 nM T00140 C32OZT 10646090 IC50 = 100 nM T00140 CY83LZ 10646383 IC50 = 20 nM T00140 C7SAB5 10646479 IC50 = 140 nM T00140 CM6CN8 10646537 IC50 = 820 nM T00140 CN0KH9 10647043 IC50 = 20 nM T00140 CIY8X1 10647748 IC50 = 10 nM T00140 CKOM02 10649058 IC50 = 23 nM T00140 C9ZS3M 10649059 IC50 = 21 nM T00140 C8DH4N 10651780 IC50 = 360 nM T00140 CK9I0H 10652263 IC50 = 130 nM T00140 CLJ1U5 10655329 IC50 = 2000 nM T00140 C6S8ZI 10655427 IC50 = 1000 nM T00140 COV83P 10655964 IC50 = 3500 nM T00140 C9A1HL 10656046 IC50 = 880 nM T00140 C9WFI3 10658954 IC50 = 5300 nM T00140 C9FMU7 10659698 IC50 = 1500 nM T00140 C3K6VD 10660093 IC50 = 680 nM T00140 C2XCM6 10671979 IC50 = 56 nM T00140 CN4L1D 10672437 IC50 = 22 nM T00140 CWFZ95 10672718 IC50 = 48 nM T00140 C8EFB2 10675837 IC50 = 23 nM T00140 CN68KT 10679286 IC50 = 7900 nM T00140 C5W1YE 10680149 IC50 = 1700 nM T00140 CIA86R 10681296 IC50 = 1100 nM T00140 CJ2BT6 10684287 IC50 = 60 nM T00140 CD1N4Z 10686077 IC50 = 160 nM T00140 CF21EA 10694045 IC50 = 70 nM T00140 C90FKN 10697771 IC50 = 2215 nM T00140 C7JKO8 10702459 IC50 = 8600 nM T00140 C69YPB 10704214 IC50 = 4800 nM T00140 CC80OZ 10706217 IC50 = 3600 nM T00140 CDPT71 10709447 IC50 = 12000 nM T00140 CZ8RA0 10716389 IC50 = 143 nM T00140 CJX4U3 10717163 IC50 = 490 nM T00140 C62WKD 10718706 IC50 = 40 nM T00140 CW7HZ2 10720814 IC50 = 20 nM T00140 C8CU4E 10722510 IC50 = 52 nM T00140 C8YH7S 10725595 IC50 = 1800 nM T00140 CP5QF4 10725826 IC50 = 460 nM T00140 C4EQP6 10725868 IC50 = 900 nM T00140 CRF0S3 10726150 IC50 = 380 nM T00140 C6TXQ0 10726208 IC50 = 1800 nM T00140 CIU76E 10726380 IC50 = 5800 nM T00140 CD25MI 10726535 IC50 = 760 nM T00140 CP97JR 10726930 IC50 = 3800 nM T00140 COK6J8 10726964 IC50 = 1700 nM T00140 CL5XI2 10729662 IC50 = 1600 nM T00140 C39DJY 10729840 IC50 = 8400 nM T00140 CR06ZW 10739259 IC50 = 52 nM T00140 C0A7BD 10741398 IC50 = 27 nM T00140 CUP96L 10741947 IC50 = 426 nM T00140 C2MU5E 10742029 IC50 = 30 nM T00140 C7OLQ0 10742030 IC50 = 13 nM T00140 CSC18B 10742031 IC50 = 29 nM T00140 C10ETF 10746661 IC50 = 175 nM T00140 CRL7P5 10749417 IC50 = 740 nM T00140 C2RF7V 10751689 IC50 = 2700 nM T00140 CBX61V 10754395 IC50 = 3100 nM T00140 C3PL8Z 10754558 IC50 = 2500 nM T00140 CY8LV9 10755909 IC50 = 100 nM T00140 CJR19I 10757665 IC50 = 10000 nM T00140 CLX3B8 10761531 IC50 = 150 nM T00140 C0QTL8 10765188 IC50 = 18 nM T00140 CW3X7H 10766653 IC50 = 14 nM T00140 CSP05M 10766748 IC50 = 21 nM T00140 CC80DW 10767794 IC50 = 17 nM T00140 CB1T4Y 10768311 IC50 = 120 nM T00140 CA8J5Q 10770349 IC50 = 100 nM T00140 CIC64P 10770666 IC50 = 30 nM T00140 CT9M0K 10774258 IC50 = 160 nM T00140 CFT3H1 10776511 IC50 = 3600 nM T00140 C80GDN 10779627 IC50 = 2600 nM T00140 C9XMZ2 10781788 IC50 = 150 nM T00140 CQ5XW6 10786611 IC50 = 142 nM T00140 CR6KC4 10788213 IC50 = 25 nM T00140 CJ29TP 10790769 IC50 = 14 nM T00140 CZNK34 10794157 IC50 = 70 nM T00140 CKB8C4 10797495 IC50 = 440 nM T00140 CT14RN 10798098 IC50 = 430 nM T00140 CD1JN4 10798630 IC50 = 4600 nM T00140 CJA5X1 10798906 IC50 = 1500 nM T00140 C9Q1VF 10799877 IC50 = 520 nM T00140 C2G3CQ 10801450 IC50 = 1400 nM T00140 C3G5JB 10802123 IC50 = 140 nM T00140 CK15ZJ 10812930 IC50 = 60 nM T00140 C20UNG 10814786 IC50 = 9 nM T00140 CE1A2M 10818116 IC50 = 62 nM T00140 CIYU17 10820552 IC50 = 1000 nM T00140 C7TPG5 10821903 IC50 = 4100 nM T00140 C3O1SB 10822291 IC50 = 1800 nM T00140 C8REX5 10822398 IC50 = 2100 nM T00140 CV8RN3 10823449 IC50 = 600 nM T00140 C1GOU9 10824904 IC50 > 50000 nM T00140 CP23RJ 10825845 IC50 = 2600 nM T00140 C32UVY 10826834 IC50 = 200 nM T00140 C6S9VL 10827210 IC50 = 1600 nM T00140 C27IXS 10834151 IC50 = 360 nM T00140 CRI9P2 10834926 IC50 = 1000 nM T00140 C0C5AY 10842086 IC50 = 170 nM T00140 CYDB70 10842207 IC50 = 60 nM T00140 C91VZI 10845542 IC50 = 3000 nM T00140 CKMB23 10845994 IC50 = 13000 nM T00140 CBMN58 10847424 IC50 = 23000 nM T00140 CO13DJ 10847997 IC50 = 1400 nM T00140 CUK06A 10849293 IC50 = 24000 nM T00140 CL18DH 10849702 IC50 = 3100 nM T00140 CF98BX 10850793 IC50 = 9000 nM T00140 C46JCP 10852345 IC50 = 5000 nM T00140 CK7WG2 10873133 IC50 = 1400 nM T00140 C23VDE 10999992 IC50 = 18400 nM T00140 CHT16X 11019578 IC50 = 4200 nM T00140 CL74SR 11057468 IC50 = 500 nM T00140 CBRW71 11156027 IC50 = 770 nM T00140 CW1M8Q 11160272 IC50 = 530 nM T00140 CN68EX 11164952 IC50 > 1000 nM T00140 C9KX7V 11180042 IC50 = 800 nM T00140 CU82SZ 11202736 IC50 > 10000 nM T00140 CU01PR 11213050 IC50 > 10000 nM T00140 CM5Z6L 11213438 IC50 > 10000 nM T00140 CYX84A 11213988 IC50 > 10000 nM T00140 CDH1L4 11222461 IC50 > 10000 nM T00140 CA4TQ6 11248759 IC50 > 3000 nM T00140 CD0T4Y 11259519 IC50 > 10000 nM T00140 CJ2C7K 11261258 IC50 = 850 nM T00140 CQ8T0K 11269805 IC50 = 130 nM T00140 CB76HJ 11269914 IC50 = 72 nM T00140 CPFA56 11281242 IC50 = 150 nM T00140 CY8K9F 11282341 IC50 > 10000 nM T00140 C6NI5K 11301895 IC50 > 10000 nM T00140 CX35FW 11304929 IC50 > 1000 nM T00140 C8GI1X 11315837 IC50 > 1000 nM T00140 C0NC7H 11317417 IC50 = 720 nM T00140 CF6TZ4 11329239 IC50 = 760 nM T00140 CLHA87 11339601 IC50 = 200 nM T00140 C09HXJ 11340857 IC50 = 830 nM T00140 C1UH4A 11350397 IC50 = 80 nM T00140 C1XM5N 11362777 IC50 > 1000 nM T00140 C2EJ0X 11374699 IC50 > 10000 nM T00140 CQW25D 11376787 IC50 = 72 nM T00140 CP2ID5 11386458 IC50 > 40000 nM T00140 CGQK95 11398561 IC50 = 740 nM T00140 C1ICK8 11430770 IC50 > 10000 nM T00140 CI6AL4 11442938 IC50 = 480 nM T00140 C6RG5B 11466350 IC50 > 10000 nM T00140 CZ40LW 11487048 IC50 = 280 nM T00140 CD43NT 11487702 IC50 > 10000 nM T00140 CXU3T1 11487950 IC50 = 570 nM T00140 CZ24YQ 11500329 IC50 = 2300 nM T00140 CH8KJ1 11500409 IC50 = 7100 nM T00140 CM2GL9 11530031 IC50 = 300 nM T00140 C2S3LP 11530690 IC50 = 3100 nM T00140 CCX16G 11532986 IC50 = 3500 nM T00140 CO8LJ4 11592681 IC50 = 980 nM T00140 CYFB38 11596459 IC50 = 2300 nM T00140 CRPF12 11602022 IC50 = 5000 nM T00140 C8JFC6 11637678 IC50 = 2800 nM T00140 CUEB81 11645226 IC50 = 9700 nM T00140 CO20UA 11674232 IC50 = 1200 nM T00140 C8PJ6B 11677372 IC50 > 3000 nM T00140 C80FMB 11742136 IC50 > 10000 nM T00140 C0A4JW 11774961 IC50 = 810 nM T00140 C8RG2P 11779569 IC50 = 4000 nM T00140 C95GBO 11796680 IC50 = 15 nM T00140 C26BMJ 11799138 IC50 = 67 nM T00140 C2D1SV 11799384 IC50 = 31 nM T00140 CHU8W2 11802470 IC50 = 60 nM T00140 CVT0F8 11808877 IC50 = 420 nM T00140 C0VC7D 11834888 IC50 = 5300 nM T00140 CQ2XI6 11837345 IC50 = 8000 nM T00140 C3GD7O 11856170 IC50 = 65 nM T00140 CSX4C0 11866208 IC50 = 900 nM T00140 CBE30L 11962168 IC50 = 17000 nM T00140 CJO9Z6 11978569 IC50 = 5000 nM T00140 C63RLZ 11983343 IC50 = 2100 nM T00140 C83XGW 12297476 IC50 = 4710 nM T00140 CPKA02 12305221 IC50 > 40000 nM T00140 CJ65IL 12305517 IC50 = 42000 nM T00140 CKNP83 12309637 IC50 = 13800 nM T00140 C0X1AE 12310283 IC50 = 25700 nM T00140 CKI97Z 12344252 IC50 > 200000 nM T00140 CVP30J 12395137 IC50 = 450 nM T00140 CKSL53 12507616 IC50 > 200000 nM T00140 CK08CX 12533628 IC50 = 4600 nM T00140 CTQ31G 12658321 IC50 = 2900 nM T00140 CELM69 12801541 IC50 = 31800 nM T00140 CB9G2Y 12992627 IC50 = 194 nM T00140 CWOJ46 12992629 IC50 = 57 nM T00140 COF8W3 13008156 IC50 > 200000 nM T00140 CH9VC8 13245625 IC50 > 1000 nM T00140 CKZ09L 13592040 IC50 = 130 nM T00140 CS2HW8 13592041 IC50 = 63 nM T00140 CQ1F5K 13592042 IC50 = 59 nM T00140 C3OJ0X 13592043 IC50 = 170 nM T00140 C1T6SK 13592044 IC50 = 220 nM T00140 C5HYO4 13592047 IC50 = 71 nM T00140 C0LR8A 13592053 IC50 = 290 nM T00140 CQO57E 13592057 IC50 = 520 nM T00140 CLW17Z 13670402 IC50 = 130 nM T00140 C4UF6B 13833994 IC50 = 270 nM T00140 C0P5AK 13914227 IC50 = 2400 nM T00140 C49OGE 13914253 IC50 = 19600 nM T00140 C0LB6O 13918608 IC50 > 50000 nM T00140 C9ETH1 13974499 IC50 = 2200 nM T00140 C4U3RD 14006855 IC50 = 50 nM T00140 C5J0PE 14167253 IC50 = 30600 nM T00140 C5LH9S 14213209 IC50 = 41400 nM T00140 CZUI98 14213211 IC50 = 27200 nM T00140 C0GLC7 14213215 IC50 > 50000 nM T00140 CIT35C 14213224 IC50 > 50000 nM T00140 C6EZ0K 14312565 IC50 > 1000 nM T00140 C5KF2O 14376458 IC50 = 250 nM T00140 CKS1X0 14406193 IC50 = 120 nM T00140 CG10ZI 14406194 IC50 = 100 nM T00140 C7X4BJ 14406195 IC50 = 2000 nM T00140 C0P2EA 14406197 IC50 = 600 nM T00140 CX59IP 14406199 IC50 = 130 nM T00140 CU2J6V 14406200 IC50 = 30 nM T00140 COTI07 14406201 IC50 = 3000 nM T00140 CI3X2N 14406202 IC50 = 1000 nM T00140 CC5L8H 14406203 IC50 = 1000 nM T00140 C07PJE 14406204 IC50 = 1300 nM T00140 C7XS8Y 14406209 IC50 = 1200 nM T00140 CK5DM3 14406212 IC50 = 100 nM T00140 C4VCA8 14406214 IC50 = 250 nM T00140 C82ITK 14406216 IC50 = 160 nM T00140 C5L4XD 14406218 IC50 = 2500 nM T00140 C2X8PQ 14416570 IC50 = 1200 nM T00140 C5PT1G 14416572 IC50 2700 nM T00140 C1SG0F 14416576 IC50 > 1000 nM T00140 CRYI80 14416580 IC50 > 1000 nM T00140 C27NOS 14416585 IC50 = 200 nM T00140 C6BP2F 14416587 IC50 < 1000 nM T00140 CS1XR2 14448070 IC50 > 200000 nM T00140 CX8O1D 14545016 IC50 = 500 nM T00140 CO5VF3 14545017 IC50 = 4000 nM T00140 C19VLP 14545020 IC50 = 250 nM T00140 CH7KD8 14545024 IC50 = 50 nM T00140 CD73NH 14545025 IC50 = 100 nM T00140 CN6R3M 14545026 IC50 < 10000 nM T00140 C27NKC 14545027 IC50 = 300 nM T00140 CKT7O5 14570888 IC50 = 574 nM T00140 CI90ER 14570889 IC50 = 31 nM T00140 C7VZR3 14570890 IC50 = 860 nM T00140 C0X5KJ 14570891 IC50 = 99 nM T00140 C8UFW4 14570892 IC50 = 7 nM T00140 CXT93P 14570893 IC50 = 20 nM T00140 C6VDH7 14570894 IC50 = 30 nM T00140 CKO8G2 14570895 IC50 = 26 nM T00140 CSJ82A 14570896 IC50 = 13 nM T00140 C41YSN 14570899 IC50 = 12 nM T00140 CX6V5H 14570900 IC50 = 376 nM T00140 CUF1Q0 14570903 IC50 = 46 nM T00140 COAD07 14570904 IC50 = 291 nM T00140 CK72SD 14570905 IC50 = 20 nM T00140 CC56YI 14570907 IC50 = 76 nM T00140 C3UD2O 14570908 IC50 = 2134 nM T00140 C76PXO 14570914 IC50 = 105 nM T00140 C7VH5T 14576502 IC50 = 6000 nM T00140 CW5ZQ1 14761244 IC50 = 760000 nM T00140 C4PS0F 14771889 IC50 ~ 100 nM T00140 CV41BE 14771890 IC50 = 86 nM T00140 CCX7K5 14771891 IC50 = 90 nM T00140 CG57JP 14771892 IC50 = 86 nM T00140 C91VJM 14771893 IC50 < 1000 nM T00140 C0EMA5 14771894 IC50 < 1000 nM T00140 CZ4WJ2 14771895 IC50 = 65 nM T00140 CV5YH8 14771896 IC50 < 1000 nM T00140 C3HNQ2 14771897 IC50 ~ 100 nM T00140 CH0TC9 14771898 IC50 < 1000 nM T00140 CX3N7Z 14771899 IC50 = 370 nM T00140 CX7VA0 14771900 IC50 > 1000 nM T00140 CZC2D4 14771901 IC50 < 1000 nM T00140 CTY60Q 14771902 IC50 < 1000 nM T00140 C0D5OC 14771903 IC50 = 91 nM T00140 CS3V5C 14771904 IC50 < 1000 nM T00140 CNH5M1 14771905 IC50 = 290 nM T00140 CXN94C 14771906 IC50 = 590 nM T00140 CY2HF8 14771907 IC50 > 1000 nM T00140 CP5M9A 14771908 IC50 < 1000 nM T00140 CI3XK7 14771909 IC50 ~ 1000 nM T00140 C8NTK2 14771910 IC50 = 170 nM T00140 C8H6XA 14771911 IC50 = 130 nM T00140 CK53TR 14771912 IC50 < 1000 nM T00140 C10DIY 14771913 IC50 < 1000 nM T00140 C2F9TX 14771915 IC50 = 100 nM T00140 C83VPQ 14771916 IC50 < 1000 nM T00140 CA0C7U 14771917 IC50 < 1000 nM T00140 CK0AR5 14771918 IC50 < 1000 nM T00140 C8SRH6 14771919 IC50 > 1000 nM T00140 CCS9Y4 14771920 IC50 > 1000 nM T00140 C47LJK 14771921 IC50 > 1000 nM T00140 C9OWP0 14771922 IC50 < 1000 nM T00140 C1Z6FX 14771923 IC50 < 1000 nM T00140 CHI8M3 14771924 IC50 = 45 nM T00140 C4JX5S 14771927 IC50 < 1000 nM T00140 CRGJ45 14771928 IC50 < 1000 nM T00140 C7L2ZJ 14771929 IC50 < 1000 nM T00140 CXAG49 14771930 IC50 > 1000 nM T00140 C54ITL 14771931 IC50 < 1000 nM T00140 CC4LM1 14771932 IC50 > 1000 nM T00140 CU6TO3 14771933 IC50 > 1000 nM T00140 C08CRZ 14771934 IC50 = 430 nM T00140 CA3D5U 14771935 IC50 < 1000 nM T00140 CZU2H5 14771936 IC50 > 1000 nM T00140 C3B0LX 14771937 IC50 > 1000 nM T00140 CRT9E4 14771938 IC50 > 1000 nM T00140 CIK71M 14836119 IC50 = 800 nM T00140 CWM83A 14845590 IC50 > 10000 nM T00140 C7AC2F 14873670 IC50 = 800 nM T00140 CV9WO2 14873671 IC50 = 100 nM T00140 CR94OG 14873672 IC50 = 58 nM T00140 C4FVN8 14873673 IC50 = 62 nM T00140 C1U9XH 14873674 IC50 = 86 nM T00140 C3PM7U 14873675 IC50 = 105 nM T00140 CUJL79 14873676 IC50 = 115 nM T00140 CEU34W 14873677 IC50 = 500 nM T00140 C7N5MW 14873678 IC50 = 1400 nM T00140 C4XD6P 14873679 IC50 = 500 nM T00140 CWK51O 14873680 IC50 = 220 nM T00140 CL5HF2 14873681 IC50 = 250 nM T00140 C76QVC 14873682 IC50 = 190 nM T00140 CUV86G 14873683 IC50 = 175 nM T00140 CL1G9F 14873684 IC50 = 240 nM T00140 C2K5ZS 14873685 IC50 = 950 nM T00140 CCV2P9 14873686 IC50 = 300 nM T00140 CE2C3P 14873687 IC50 = 115 nM T00140 CU8S5Z 14873688 IC50 = 115 nM T00140 C01ZNY 14873689 IC50 = 140 nM T00140 C1GE7P 14873690 IC50 = 135 nM T00140 CMW5V0 14873691 IC50 = 340 nM T00140 C4KGB9 14873692 IC50 = 500 nM T00140 CZS0J3 14873693 IC50 = 1500 nM T00140 C0CZ5P 14873694 IC50 = 480 nM T00140 CZ3Y1E 14873695 IC50 = 265 nM T00140 C0XBO2 14873696 IC50 = 110 nM T00140 CXE61G 14873697 IC50 = 155 nM T00140 CT9Y0K 14873698 IC50 = 270 nM T00140 C87HJA 14873699 IC50 = 210 nM T00140 C4OJ3I 14873700 IC50 = 870 nM T00140 C4MEP2 14873701 IC50 = 1250 nM T00140 C91BUN 14873707 IC50 = 88 nM T00140 CA91TP 14873708 IC50 = 128 nM T00140 CZO9W4 14873709 IC50 = 350 nM T00140 CR94AQ 14873710 IC50 = 770 nM T00140 CR3D4S 14873716 IC50 = 126 nM T00140 CN1WY6 14873717 IC50 = 280 nM T00140 C5UTX2 14873718 IC50 = 480 nM T00140 C6EU8P 14873719 IC50 = 1350 nM T00140 CZY58X 14898748 IC50 = 300 nM T00140 C3GA2F 14898751 IC50 = 300 nM T00140 C7QY8L 14898753 IC50 = 1500 nM T00140 CFI5J9 14971254 IC50 = 180 nM T00140 CIX50A 14971255 IC50 = 400 nM T00140 CRAM53 14971256 IC50 = 100 nM T00140 CMK7S5 14971277 IC50 = 3600 nM T00140 CYN8P3 14971278 IC50 = 380 nM T00140 C5LYB8 14971279 IC50 = 430 nM T00140 C2JMC3 14971280 IC50 = 280 nM T00140 C2QME7 14971281 IC50 = 1390 nM T00140 CBK4Q5 14971282 IC50 = 130 nM T00140 CBQ17Z 14971283 IC50 = 42 nM T00140 C16TZW 14971284 IC50 = 1900 nM T00140 C32RLZ 14971285 IC50 = 180 nM T00140 CK1LW7 14971286 IC50 = 36 nM T00140 C8WKT5 14971287 IC50 = 24 nM T00140 CJW8U5 14971289 IC50 = 63 nM T00140 C0GT3E 14971290 IC50 = 65 nM T00140 CQ6Z9F 14971291 IC50 = 4400 nM T00140 CG62YT 14971292 IC50 = 240 nM T00140 C3QRS5 14971293 IC50 = 440 nM T00140 C14DEI 14971294 IC50 = 37 nM T00140 CUP6B8 14971295 IC50 = 74 nM T00140 CFZ48U 14971296 IC50 = 86 nM T00140 C4DSH5 14971300 IC50 = 310 nM T00140 C10VPI 14971301 IC50 = 1400 nM T00140 C0A7QB 14971302 IC50 = 240 nM T00140 CUJ9F0 14971308 IC50 = 220 nM T00140 CJ5HX7 14971309 IC50 = 120 nM T00140 CY65UM 14971310 IC50 = 880 nM T00140 CZ5FM1 14971311 IC50 = 320 nM T00140 C30QTK 14971312 IC50 = 310 nM T00140 C93DKA 14971314 IC50 = 200 nM T00140 CUR18K 14971315 IC50 = 53 nM T00140 CXE6O5 14971318 IC50 > 3000 nM T00140 C4HKJ7 14980538 IC50 = 165 nM T00140 COB0M4 14980539 IC50 = 35 nM T00140 C4A2JX 14980540 IC50 = 27 nM T00140 CRBN10 14980541 IC50 = 80 nM T00140 C98AEV 14980542 IC50 = 12 nM T00140 CY5H7I 14980543 IC50 = 66 nM T00140 C7SVF6 14980544 IC50 = 42 nM T00140 C6OFC1 14980546 IC50 = 3 nM T00140 C3OR9Q 14980547 IC50 = 20 nM T00140 CM6VZ9 14980548 IC50 = 28 nM T00140 C6UN3B 14980553 IC50 = 500 nM T00140 C7BVF6 14980554 IC50 = 300 nM T00140 CU89MF 14980555 IC50 = 95 nM T00140 CI31GS 14980556 IC50 = 23 nM T00140 C8C9LB 14980557 IC50 = 33 nM T00140 CXWJ92 14980558 IC50 = 110 nM T00140 CO0U1F 14980559 IC50 = 16 nM T00140 CNH08B 14980560 IC50 = 28 nM T00140 CRF26H 14980561 IC50 = 28 nM T00140 CH0R4U 14980563 IC50 = 420 nM T00140 CDN75W 14980566 IC50 = 170 nM T00140 CST6Y8 14980570 IC50 = 100 nM T00140 C7H9RS 14980579 IC50 = 88 nM T00140 CO6LG2 14980582 IC50 = 33 nM T00140 C4R7GX 14980586 IC50 = 210 nM T00140 C7SZL6 14980593 IC50 = 97 nM T00140 CC6I4H 14980594 IC50 = 38 nM T00140 C1YR7N 14980595 IC50 = 23 nM T00140 C0J6DC 14980600 IC50 = 12 nM T00140 CFVH72 14980601 IC50 = 19 nM T00140 C2FXV4 14980604 IC50 = 11 nM T00140 CZNM37 14980605 IC50 = 125 nM T00140 C65OLS 14985863 IC50 > 40000 nM T00140 C3HBZ7 14985864 IC50 = 400 nM T00140 CL1S0J 14985865 IC50 = 4200 nM T00140 CY45LU 14985866 IC50 = 10600 nM T00140 CYVW67 14985869 IC50 = 300 nM T00140 CR54PD 14985873 IC50 = 600 nM T00140 CY98EZ 14985877 IC50 = 200 nM T00140 CZ38NR 14985893 IC50 = 2500 nM T00140 CHK1O8 14985894 IC50 = 1700 nM T00140 CRWH93 14985895 IC50 = 700 nM T00140 C3UH7B 14985897 IC50 = 2500 nM T00140 CZHT08 14985898 IC50 = 2600 nM T00140 CM2WU6 14985899 IC50 = 19000 nM T00140 C92MLN 14985900 IC50 = 600 nM T00140 C9X7GB 14985901 IC50 = 40000 nM T00140 CS21VM 14985910 IC50 = 70 nM T00140 CG4JR8 14985911 IC50 = 400 nM T00140 C87SUY 14985912 IC50 = 200 nM T00140 CF0D4Y 14985914 IC50 = 200 nM T00140 CCT65A 14985915 IC50 = 400 nM T00140 COW68H 14985916 IC50 = 30 nM T00140 CTZ61U 14985917 IC50 = 1300 nM T00140 C1YV7X 14985918 IC50 = 200 nM T00140 CLQ2J9 14985919 IC50 = 300 nM T00140 CK9F2N 14985920 IC50 = 80 nM T00140 C7Y0SA 14985921 IC50 = 200 nM T00140 CFL2B0 14985922 IC50 = 40 nM T00140 CB3KM4 14985923 IC50 = 50 nM T00140 C2PE4Q 15005943 EC50 = 39 nM T00140 C1T8NI 15005945 EC50 = 20 nM T00140 C09GIO 15005946 EC50 = 70 nM T00140 CZR39X 15005948 EC50 = 130 nM T00140 C0LO5Q 15005961 EC50 = 90 nM T00140 CM0V7I 15005962 EC50 = 130 nM T00140 C78ZXU 15005966 EC50 = 110 nM T00140 CO3BH4 15005967 EC50 = 1070 nM T00140 C9K3GS 15005968 EC50 = 20 nM T00140 C5S2MP 15005969 EC50 = 70 nM T00140 C3SQ7B 15005970 EC50 = 390 nM T00140 C40AHT 15005971 EC50 = 5200 nM T00140 C21ZUJ 15005972 EC50 = 24500 nM T00140 CDNE23 15005973 EC50 = 45 nM T00140 CAKD61 15005974 EC50 = 3200 nM T00140 CDP6E0 15005975 EC50 = 530 nM T00140 C2R9GF 15005976 EC50 = 160 nM T00140 C1GV0Q 15005977 EC50 = 70 nM T00140 CUN53P 15049958 IC50 ~ 40000 nM T00140 CMT17N 15049978 IC50 = 900 nM T00140 CF8OB6 15049981 IC50 = 7600 nM T00140 C4GUL8 15049985 IC50 > 40000 nM T00140 C7RPG4 15049987 IC50 = 4800 nM T00140 C5VF2R 15049997 IC50 ~ 40000 nM T00140 CT79OQ 15049998 IC50 ~ 40000 nM T00140 C0JE3M 15050004 IC50 = 7000 nM T00140 CUG96T 15050005 IC50 = 500 nM T00140 CHDV56 15050006 IC50 > 40000 nM T00140 C0H3LV 15050007 IC50 ~ 40000 nM T00140 C3C9ZN 15050008 IC50 = 600 nM T00140 C7GZL6 15050009 IC50 = 6300 nM T00140 C97QUI 15050015 IC50 = 40000 nM T00140 CGO96H 15050017 IC50 = 6300 nM T00140 C6ZDX8 15050019 IC50 = 7000 nM T00140 CD8K2O 15056509 IC50 = 9300 nM T00140 CHK51C 15056510 IC50 = 6700 nM T00140 CRY03A 15056511 IC50 = 156000 nM T00140 CX5S9L 15056514 IC50 = 5200 nM T00140 CZS28R 15056515 IC50 = 39000 nM T00140 CLD4A1 15056516 IC50 = 3000 nM T00140 C9PY1F 15056517 IC50 = 125000 nM T00140 CCG1W6 15056522 IC50 = 5600 nM T00140 CI5HL4 15056537 IC50 = 3400 nM T00140 CLTJ42 15056538 IC50 = 57000 nM T00140 CM9UY6 15056539 IC50 = 277000 nM T00140 CLM52R 15056540 IC50 = 99000 nM T00140 C7GYA5 15056541 IC50 = 2500 nM T00140 CX82ZI 15056542 IC50 = 79000 nM T00140 CCHP75 15056543 IC50 = 1800 nM T00140 CS46EO 15153337 IC50 = 6000 nM T00140 C4L7PE 15181201 IC50 > 40000 nM T00140 CUB5N8 15199688 IC50 = 75 nM T00140 C2KVM1 15283092 IC50 = 26 nM T00140 CI7P3D 15283094 IC50 = 720 nM T00140 CIXJ84 15283095 IC50 = 280 nM T00140 CV3G0M 15283097 IC50 = 27 nM T00140 CHN0O9 15379534 IC50 = 2500 nM T00140 CHOU39 15407872 IC50 = 100 nM T00140 C9AZX3 15496169 IC50 > 50000 nM T00140 C19GJV 15549539 IC50 = 600 nM T00140 CPR35F 15558820 IC50 = 250 nM T00140 C5B1IH 15560324 IC50 > 40000 nM T00140 CBD45Z 15637380 IC50 = 10 nM T00140 C1LMP9 15691787 IC50 = 470 nM T00140 CKE20P 15691788 IC50 = 740 nM T00140 C8Z6VM 15691790 IC50 = 2900 nM T00140 C7H4JT 15691798 IC50 = 5100 nM T00140 CZ1J3H 15691801 IC50 = 4500 nM T00140 CZ5VX4 15780544 IC50 = 48 nM T00140 CI1EC9 16068009 IC50 = 55 nM T00140 CN6O1U 16068119 IC50 = 40 nM T00140 C3ZKJ5 16068120 IC50 = 11 nM T00140 CPLU48 16068121 IC50 = 88 nM T00140 C9S6QP 16068233 IC50 = 19 nM T00140 CB9Z0L 16068234 IC50 = 198 nM T00140 CW4U7H 16068235 IC50 = 263 nM T00140 CT4JA5 16068236 IC50 = 1890 nM T00140 C8SQ5I 16068237 IC50 = 260 nM T00140 C28FGO 16093504 IC50 = 1900 nM T00140 C03ETJ 16681478 IC50 = 5600 nM T00140 CCPS15 16753427 IC50 = 34000 nM T00140 CKE41X 16753429 IC50 = 1500 nM T00140 C7M5CP 16753431 IC50 = 31000 nM T00140 CN8WX3 16757526 IC50 = 1220 nM T00140 CK08XF 17600320 IC50 = 82000 nM T00140 CWC71F 17865655 IC50 = 4600 nM T00140 C5HW9J 17968847 IC50 = 2200 nM T00140 C07YED 18771446 IC50 = 550 nM T00140 CHG08W 18771451 IC50 = 590 nM T00140 C7A5SQ 18771453 IC50 = 1140 nM T00140 CG70VX 18771471 IC50 = 270 nM T00140 C0CHV4 18771498 IC50 = 500 nM T00140 CVTS42 18771530 IC50 = 120 nM T00140 C24MFJ 18771532 IC50 = 120 nM T00140 CYL4X7 18771545 IC50 = 200 nM T00140 CM2LG7 18771550 IC50 = 80 nM T00140 CPR3V1 18771558 IC50 = 2300 nM T00140 CSG5A6 18771560 IC50 = 710 nM T00140 C4TD3O 18771561 IC50 = 50 nM T00140 C3Q4YM 18771574 IC50 > 5000 nM T00140 CYLR21 18786349 IC50 > 1000 nM T00140 CE39BT 18786356 IC50 = 270 nM T00140 CCP6S0 18786367 IC50 = 140 nM T00140 C81DIY 19080640 IC50 = 1300 nM T00140 CX8YE7 19349871 IC50 > 1000 nM T00140 C93XRU 19353391 IC50 = 4200 nM T00140 C1HJ5C 19756612 IC50 = 350 nM T00140 CGU69S 19773051 IC50 = 8800 nM T00140 C4V1IS 19773052 IC50 = 5100 nM T00140 C1HMD9 19894204 IC50 = 1200 nM T00140 CEU72O 19894212 IC50 = 900 nM T00140 CM3S4Z 19894214 IC50 = 230 nM T00140 CIMX82 19894227 IC50 = 970 nM T00140 C5PKJ0 19894247 IC50 = 150 nM T00140 C89VBR 19894263 IC50 = 1100 nM T00140 C89PVS 20055661 IC50 > 40000 nM T00140 CS51IE 20080675 IC50 = 200 nM T00140 CKY1V4 20376778 IC50 > 50000 nM T00140 C40UHL 21476400 IC50 > 5000 nM T00140 CLS5X8 21847229 IC50 > 8000 nM T00140 CC8JY4 22496401 IC50 = 600 nM T00140 C5LM6C 23176602 IC50 = 380 nM T00140 C2MJU1 23381046 IC50 = 90 nM T00140 C2XRV0 23546056 IC50 = 4100 nM T00140 C5Z4BD 23624475 IC50 = 2000 nM T00140 CGV7U5 23646340 IC50 = 380 nM T00140 C3BFI7 23680513 IC50 = 34 nM T00140 CSYH13 24043496 IC50 = 15000 nM T00140 C4B5MX 24824762 IC50 = 60 nM T00140 C9DO6A 24825393 IC50 > 10000 nM T00140 CK7M8I 24825399 IC50 = 8900 nM T00140 CFN79S 24825402 IC50 > 3000 nM T00140 CQK5S6 24825412 IC50 > 10000 nM T00140 CW51RK 24828806 IC50 = 3900 nM T00140 CCD95H 24854123 IC50 = 380 nM T00140 C4IP5C 24871714 IC50 = 2600 nM T00140 C7CZA0 24894101 IC50 = 10000 nM T00140 C38YDW 24971271 IC50 = 2600 nM T00140 C9F0AN 24971272 IC50 = 3200 nM T00140 CB8L5V 24971273 IC50 = 1800 nM T00140 C1IU7P 24971274 IC50 = 1200 nM T00140 CKS85U 24971275 IC50 = 1100 nM T00140 C2F9XY 24971276 IC50 = 600 nM T00140 CXIB21 24971277 IC50 = 1700 nM T00140 C5Z1YK 24971278 IC50 = 1400 nM T00140 C7Y4GR 25058073 IC50 = 3100 nM T00140 CXH48N 25058075 IC50 = 1300 nM T00140 CU1C6R 25100738 IC50 = 30 nM T00140 C1WQ7F 25141098 IC50 = 900 nM T00140 CGW49I 25146686 IC50 > 200000 nM T00140 C6RZC2 25147690 IC50 = 1000 nM T00140 C0PAE1 25179516 IC50 = 7600 nM T00140 C5RBW3 25179712 IC50 = 1500 nM T00140 CL3Q7B 25179713 IC50 = 1500 nM T00140 C54DIT 25179907 IC50 = 600 nM T00140 C9GB6J 25179909 IC50 = 700 nM T00140 CC9N3E 25179911 IC50 = 500 nM T00140 CUTK18 25179912 IC50 = 800 nM T00140 CAVM57 25187677 IC50 = 2400 nM T00140 C15RWA 25801821 IC50 = 1530 nM T00140 CY3ER7 26368018 IC50 = 300 nM T00140 CYZ6B0 26389403 IC50 > 50000 nM T00140 C46PZG 42609834 IC50 = 30 nM T00140 C1YPW8 42618003 IC50 > 100000 nM T00140 C4XG8L 42637235 IC50 = 7200 nM T00140 CWDY48 42637527 IC50 = 8100 nM T00140 CY4CX1 44157329 IC50 = 240 nM T00140 CH4QJ0 44157331 IC50 = 5500 nM T00140 C3GAC2 44157396 IC50 > 10000 nM T00140 CFP8C9 44157479 IC50 = 1700 nM T00140 CO04ZN 44157480 IC50 = 700 nM T00140 C2XHQ6 44157481 IC50 = 1700 nM T00140 CZ4FI2 44157482 IC50 = 5500 nM T00140 CV7CF8 44157483 IC50 = 97 nM T00140 C3QHZ6 44157484 IC50 = 500 nM T00140 CXC80L 44157553 IC50 = 95 nM T00140 CT7CM3 44157554 IC50 = 650 nM T00140 C97ING 44157555 IC50 = 67 nM T00140 C45HMZ 44157556 IC50 = 49 nM T00140 CYZ42T 44157557 IC50 = 650 nM T00140 C2S1HZ 44157558 IC50 = 9800 nM T00140 C8Z7AS 44157559 IC50 = 3500 nM T00140 CHSI97 44157630 IC50 > 30000 nM T00140 C9ET7K 44157721 IC50 = 1700 nM T00140 C76KPA 44157722 IC50 = 4800 nM T00140 CAX17B 44157723 IC50 = 2100 nM T00140 CFK07P 44157724 IC50 = 700 nM T00140 CU5IN7 44157725 IC50 = 86 nM T00140 CUGY90 44157824 IC50 = 84 nM T00140 CYIX03 44157825 IC50 = 140 nM T00140 CH59LF 44157826 IC50 = 150 nM T00140 CTA48Z 44157827 IC50 = 130 nM T00140 CIT61Z 44157828 IC50 = 1700 nM T00140 CY29SV 44157829 IC50 = 45 nM T00140 CKQ8F3 44157830 IC50 = 31 nM T00140 CPW4T9 44157926 IC50 = 130 nM T00140 CL46VN 44157927 IC50 = 130 nM T00140 C6OL1R 44157928 IC50 = 480 nM T00140 CLP20K 44157929 IC50 = 7000 nM T00140 C3AH1R 44157930 IC50 = 580 nM T00140 C9V8UX 44158011 IC50 = 7900 nM T00140 C7NZ4V 44158014 IC50 = 3400 nM T00140 CJ6I1D 44158015 IC50 > 30000 nM T00140 CC3AM0 44176135 IC50 = 2400 nM T00140 CHA7R9 44176136 IC50 = 1200 nM T00140 C3X1OB 44176137 IC50 = 330 nM T00140 C2AV1K 44190762 IC50 = 1640 nM T00140 C0EPN7 44241601 IC50 = 1000 nM T00140 CAY5U9 44241602 IC50 = 2100 nM T00140 C98GDR 44249905 IC50 = 1100 nM T00140 CT3ZF5 44255843 IC50 = 680 nM T00140 CY3NX9 44255873 IC50 = 740 nM T00140 C3OA7C 44268054 IC50 = 35 nM T00140 C37OBU 44268055 IC50 = 85 nM T00140 CC07UN 44268056 IC50 = 87 nM T00140 CGI7B3 44268061 IC50 = 2800 nM T00140 C2B9XG 44268063 IC50 = 65 nM T00140 C1YQ0R 44268064 IC50 = 1200 nM T00140 C3UK9Q 44268066 IC50 = 250 nM T00140 CL6SQ4 44268068 IC50 = 420 nM T00140 CRBQ75 44268069 IC50 = 770 nM T00140 CZ2JH7 44271197 IC50 = 3900 nM T00140 C5UDN3 44271328 IC50 = 680 nM T00140 C9GP6N 44271334 IC50 = 2770 nM T00140 C76DXA 44271370 IC50 = 6800 nM T00140 CFN51S 44271389 IC50 = 740 nM T00140 CK2NI0 44271394 IC50 = 440 nM T00140 CAV1Z5 44271424 IC50 = 430 nM T00140 CO2HK5 44271457 IC50 = 420 nM T00140 C17OZU 44271462 IC50 = 4320 nM T00140 C1C4PF 44271499 IC50 = 1320 nM T00140 CJBI60 44271973 IC50 = 100000 nM T00140 C9P6MJ 44273900 IC50 = 500 nM T00140 CD8PU2 44274196 IC50 > 40000 nM T00140 C80YHO 44274224 IC50 > 40000 nM T00140 CNX7I6 44274250 IC50 = 510 nM T00140 CLXJ08 44276989 IC50 = 204000 nM T00140 C2H7EU 44277141 IC50 = 19000 nM T00140 CV1P7M 44277240 IC50 = 6000 nM T00140 CLI64C 44277241 IC50 = 23000 nM T00140 CSUO90 44281455 IC50 = 860 nM T00140 C37RQO 44301833 IC50 = 590 nM T00140 CIGP85 44301906 IC50 = 710 nM T00140 CT39YE 44301972 IC50 = 1400 nM T00140 CSC73L 44302098 IC50 = 640 nM T00140 C0B1FM 44302302 IC50 = 830 nM T00140 CO19YB 44302311 IC50 = 90 nM T00140 CV27YU 44305166 IC50 = 420 nM T00140 C59HEB 44305175 IC50 = 450 nM T00140 C5ETY8 44305184 IC50 = 160 nM T00140 CG9BK5 44305198 IC50 > 4000 nM T00140 CE7Z9J 44305199 IC50 = 1400 nM T00140 C8Q1OX 44305234 IC50 = 380 nM T00140 C19CRS 44305243 IC50 = 42 nM T00140 C4L2WN 44305258 IC50 = 22 nM T00140 CXK75F 44305277 IC50 = 88 nM T00140 CD3L1B 44305358 IC50 = 3000 nM T00140 C51BOT 44305359 IC50 = 670 nM T00140 CK1ER0 44305436 IC50 = 230 nM T00140 C8N9LO 44305493 IC50 = 180 nM T00140 CK58WD 44305494 IC50 = 3800 nM T00140 C97OBQ 44308534 IC50 = 2200 nM T00140 C7QZ1Y 44308627 IC50 = 5500 nM T00140 CSR3B7 44309349 IC50 = 11000 nM T00140 CRSF17 44309358 IC50 = 40000 nM T00140 CB87TD 44309589 IC50 = 2500 nM T00140 CI6ZF8 44309590 IC50 = 600 nM T00140 C95GSZ 44309608 IC50 = 800 nM T00140 C49DJL 44309609 IC50 = 22000 nM T00140 C31VPD 44309636 IC50 = 1000 nM T00140 C03QVL 44309637 IC50 = 40000 nM T00140 CG1H7B 44309638 IC50 = 1100 nM T00140 CENZ76 44312371 IC50 = 3500 nM T00140 CAJL61 44312568 IC50 = 140 nM T00140 C04AFJ 44312705 IC50 = 1700 nM T00140 C5MOH0 44312748 IC50 = 510 nM T00140 CK9HY8 44316626 IC50 = 180 nM T00140 CU14CF 44318278 IC50 = 600 nM T00140 C7RZ8L 44318389 IC50 = 1100 nM T00140 CO95MZ 44318594 IC50 = 100 nM T00140 C95ITK 44318630 IC50 = 1000 nM T00140 C8A1CD 44318645 IC50 = 1700 nM T00140 C7RDF8 44321425 IC50 = 500 nM T00140 C50XKJ 44321940 IC50 = 200 nM T00140 CP9L0I 44322073 IC50 = 30000 nM T00140 CZYL49 44326825 IC50 = 830 nM T00140 CRY0D5 44327049 IC50 = 46 nM T00140 C0BQ1U 44327050 IC50 = 3 nM T00140 CXY1S8 44327083 IC50 = 11 nM T00140 C49NCQ 44327199 IC50 = 160 nM T00140 CL72DO 44329616 IC50 = 80 nM T00140 CR3F9L 44344532 IC50 = 6000 nM T00140 C5OU6Q 44344842 IC50 = 10000 nM T00140 C0QGP5 44344893 IC50 = 7500 nM T00140 CS57EP 44346017 IC50 = 34 nM T00140 C8AES6 44351208 IC50 = 40 nM T00140 C86DMX 44351354 IC50 = 60 nM T00140 CW14KS 44351359 IC50 = 100 nM T00140 C2YM4U 44351407 IC50 = 6930 nM T00140 CY7G1U 44351456 IC50 = 140 nM T00140 CM8GO5 44351457 IC50 = 20 nM T00140 CS3JX2 44351459 IC50 = 30 nM T00140 C84QJF 44351461 IC50 = 40 nM T00140 C5C6UX 44351479 IC50 = 20 nM T00140 CU9K2M 44351489 IC50 = 40 nM T00140 CQRH45 44351490 IC50 = 60 nM T00140 CNPT09 44351548 IC50 = 120 nM T00140 C95OHD 44351583 IC50 = 1500 nM T00140 C5UGR1 44351588 IC50 = 1200 nM T00140 C2ZSF6 44351593 IC50 = 80 nM T00140 CK84HY 44351594 IC50 = 520 nM T00140 CHU7P6 44351604 IC50 = 160 nM T00140 CR6YC7 44351606 IC50 = 3000 nM T00140 CV19OD 44351607 IC50 = 400 nM T00140 C95ZXH 44351608 IC50 = 240 nM T00140 C36IWQ 44351609 IC50 = 5500 nM T00140 CYTJ82 44351616 IC50 = 180 nM T00140 C1XJN2 44351618 IC50 = 320 nM T00140 C4XJ2F 44351622 IC50 = 130 nM T00140 CF39PJ 44351623 IC50 = 260 nM T00140 C2BAL6 44351624 IC50 = 760 nM T00140 CL9BE8 44351638 IC50 > 6000 nM T00140 C7X1RV 44351644 IC50 > 6000 nM T00140 CH7D9N 44351647 IC50 = 810 nM T00140 C35DXM 44351654 IC50 = 1300 nM T00140 CD7C6I 44351658 IC50 > 6000 nM T00140 C19DIA 44351659 IC50 = 120 nM T00140 CMIR10 44351693 IC50 = 120 nM T00140 CVOA56 44351721 IC50 = 80 nM T00140 CN6ZR9 44351729 IC50 = 140 nM T00140 C7JZ4X 44351741 IC50 = 380 nM T00140 CAFN01 44351742 IC50 = 360 nM T00140 C2E7NM 44351757 IC50 = 6000 nM T00140 CCK93H 44351758 IC50 > 6000 nM T00140 C45ITR 44351768 IC50 = 140 nM T00140 C3SNY9 44351777 IC50 = 23 nM T00140 CU8T6H 44351780 IC50 = 2200 nM T00140 CSQG54 44351793 IC50 = 70 nM T00140 C9BK7N 44351794 IC50 = 190 nM T00140 CEUW12 44351796 IC50 > 6000 nM T00140 CB8DL1 44351812 IC50 = 140 nM T00140 CAI29B 44351813 IC50 = 50 nM T00140 CRC68Z 44351822 IC50 = 50 nM T00140 C0DN6S 44351863 IC50 = 70 nM T00140 CS38DF 44351867 IC50 = 390 nM T00140 C2HL6C 44351870 IC50 = 640 nM T00140 CE5KY7 44367495 IC50 = 89 nM T00140 CS60KU 44367789 IC50 = 98 nM T00140 CX70IT 44367790 IC50 = 100 nM T00140 C6TJK9 44367797 IC50 = 180 nM T00140 CFM1S2 44368000 IC50 = 120 nM T00140 CX1CU3 44374613 IC50 = 1400 nM T00140 C6PE2I 44374983 IC50 = 160 nM T00140 C5DQ9K 44375410 IC50 = 21 nM T00140 CV76XM 44378000 IC50 = 100000 nM T00140 CXMA02 44378192 IC50 = 300 nM T00140 C84GOY 44378193 IC50 = 40000 nM T00140 CH3J8M 44378194 IC50 = 6000 nM T00140 CG0L4N 44378225 IC50 = 150 nM T00140 CRP8X5 44378301 IC50 = 28000 nM T00140 CYIV49 44378315 IC50 = 20000 nM T00140 CJIY23 44378334 IC50 = 20000 nM T00140 C9CGA2 44378335 IC50 = 3000 nM T00140 CVW20A 44378349 IC50 = 65000 nM T00140 C04FUX 44379922 IC50 = 7100 nM T00140 CU67KP 44389292 IC50 = 102 nM T00140 CU2X6H 44389293 IC50 = 90 nM T00140 CF27BX 44389301 IC50 = 176 nM T00140 CTG4C7 44389302 IC50 = 150 nM T00140 CXT7P9 44395497 IC50 = 68 nM T00140 C3QW5V 44395530 IC50 = 96 nM T00140 C7A1RD 44400781 IC50 > 1000 nM T00140 CO58IV 44400880 IC50 = 830 nM T00140 CMX3R5 44410427 IC50 = 300 nM T00140 CA4N0T 44410538 IC50 = 55 nM T00140 C4LZ5C 44410542 IC50 = 0.5 nM T00140 CH7N5M 44410587 IC50 = 1700 nM T00140 CKL7C5 44410588 IC50 = 2.7 nM T00140 C1G9XK 44410593 IC50 = 3.7 nM T00140 C3TG5P 44410711 IC50 = 4.3 nM T00140 CGH20N 44410712 IC50 = 0.8 nM T00140 CLU53R 44410718 IC50 = 0.5 nM T00140 CHG7L1 44423252 IC50 > 10000 nM T00140 CBG9N2 44423253 IC50 = 4000 nM T00140 CJ0EC5 44423254 IC50 = 900 nM T00140 C9N3RP 44423258 IC50 > 10000 nM T00140 CDT83A 44423267 IC50 = 3000 nM T00140 C7RO4U 44423268 IC50 = 900 nM T00140 C1IP9F 44423269 IC50 = 1000 nM T00140 C8VCY0 44447699 IC50 > 6300 nM T00140 C1O3TA 44447701 IC50 = 5000 nM T00140 CMVU38 44447702 IC50 > 6000 nM T00140 COE04Y 44457901 IC50 = 102 nM T00140 CQDZ60 44457902 IC50 = 36 nM T00140 CNAH32 44457918 IC50 > 3000 nM T00140 CL2ES9 44457974 IC50 = 1960 nM T00140 CW4PN8 44457975 IC50 = 1460 nM T00140 CTUA35 44458007 IC50 = 124 nM T00140 C2XZV9 44460112 IC50 > 15000 nM T00140 CNK7B4 44460114 IC50 > 30000 nM T00140 CG1I0J 44460122 IC50 > 15000 nM T00140 C7W1HI 44460123 IC50 > 30000 nM T00140 C4B0ZM 44460128 IC50 > 50000 nM T00140 C9OR2U 44460130 IC50 > 75000 nM T00140 CX4GJ6 44460139 IC50 > 75000 nM T00140 C2XWI4 44460175 IC50 > 100000 nM T00140 C0QD8O 44557858 IC50 > 150000 nM T00140 C04CGM 44558899 IC50 = 750 nM T00140 CY2D0A 44561035 IC50 = 15000 nM T00140 CUZA87 44561036 IC50 = 68000 nM T00140 CLP0D9 44587062 IC50 = 5000 nM T00140 C4LT2D 44591066 IC50 = 790 nM T00140 C08KAB 44591067 IC50 = 660 nM T00140 CAXW02 45110606 IC50 = 13000 nM T00140 CSLZ04 45267718 IC50 = 4800 nM T00140 C0R8MQ 45267726 IC50 = 1600 nM T00140 C8AXK3 45268597 IC50 = 1600 nM T00140 C6CEX5 45268605 IC50 = 1600 nM T00140 C0F7RJ 45268611 IC50 = 2000 nM T00140 C1EIF5 45269442 IC50 > 10000 nM T00140 CU91HN 45269452 IC50 = 900 nM T00140 C74OGR 45269453 IC50 > 10000 nM T00140 CI07HR 45269977 IC50 = 2200 nM T00140 C4X8NT 45270286 IC50 = 6000 nM T00140 CJC3M7 45270291 IC50 > 10000 nM T00140 CTX61C 45271105 IC50 = 8200 nM T00140 C5U8HX 45271112 IC50 = 1500 nM T00140 CR1QU8 45271974 IC50 = 9500 nM T00140 CN4ET7 45271983 IC50 = 4800 nM T00140 CH92UP 45271992 IC50 = 4800 nM T00140 C42QTW 45272810 IC50 = 5200 nM T00140 CVU12R 45272820 IC50 = 4500 nM T00140 COW52N 45273399 IC50 = 1100 nM T00140 COP75F 45273770 IC50 = 3000 nM T00140 CQ4GE9 45273780 IC50 > 10000 nM T00140 C14HXU 45783050 IC50 = 5900 nM T00140 CSG4V5 46172351 IC50 = 2490 nM T00140 C5IZ9B 46189193 IC50 = 600 nM T00140 CXA3M9 46189194 IC50 = 210 nM T00140 CTK35D 46189195 IC50 = 590 nM T00140 CN4RL1 46189196 IC50 = 270 nM T00140 CZL7E6 46189367 IC50 = 8100 nM T00140 CJX28F 46213934 IC50 = 2700 nM T00140 C2RTO6 46837638 IC50 = 2800 nM T00140 CM2K0V 46837639 IC50 = 2800 nM T00140 CRY5B0 46837640 IC50 = 800 nM T00140 CY85OT 46837641 IC50 = 1800 nM T00140 C2OP7F 46837642 IC50 = 900 nM T00140 CHJD18 46837643 IC50 = 700 nM T00140 CIH0K4 46837775 IC50 = 500 nM T00140 CP8OA1 46837776 IC50 = 7000 nM T00140 CV5ZO3 46837777 IC50 = 2200 nM T00140 CWFQ46 46837778 IC50 = 500 nM T00140 CD37LB 46837779 IC50 = 2800 nM T00140 CEPL58 46837915 IC50 = 6600 nM T00140 C89OMP 46837916 IC50 = 9300 nM T00140 C5YJS7 46837917 IC50 = 2400 nM T00140 CM3H5J 46837918 IC50 = 800 nM T00140 CKDW89 46837919 IC50 = 4000 nM T00140 CD5UE3 46837920 IC50 = 1200 nM T00140 C4S6ID 46838058 IC50 = 1200 nM T00140 CGI58K 46845031 IC50 = 59900 nM T00140 C9DRL8 46845033 IC50 = 59300 nM T00140 C48OCQ 46845035 IC50 = 109700 nM T00140 CET7R4 46866190 IC50 = 700 nM T00140 CSV51G 46866297 IC50 = 4200 nM T00140 CLS14Y 46866298 IC50 = 4500 nM T00140 C08GUA 46885478 IC50 = 500 nM T00140 CB6X5P 46885522 IC50 = 5800 nM T00140 CL92SR 46885552 IC50 = 700 nM T00140 CSU0B6 46885553 IC50 = 800 nM T00140 CC14YP 46885554 IC50 = 3100 nM T00140 CEQ10W 46885555 IC50 = 2400 nM T00140 CA78QN 46885556 IC50 = 2500 nM T00140 CPI5N2 46885589 IC50 = 2500 nM T00140 CP3EV2 46885590 IC50 = 1800 nM T00140 C7C6LI 46885591 IC50 = 500 nM T00140 C2VOW1 46898079 IC50 = 90 nM T00140 C68SVP 46906730 IC50 = 66400 nM T00140 CFL89P 46906732 IC50 = 92900 nM T00140 C0HYK2 46906734 IC50 = 39300 nM T00140 CZ1BI2 46906736 IC50 = 38000 nM T00140 CDY1P0 46906738 IC50 = 45400 nM T00140 CT39AY 46906740 IC50 = 47400 nM T00140 CTF2R8 46906742 IC50 = 81400 nM T00140 CH1ZW7 46906744 IC50 = 24600 nM T00140 C2PL3G 46927848 IC50 = 2400 nM T00140 C25VSJ 46927960 IC50 = 4000 nM T00140 CB7XA0 49788946 IC50 > 10000 nM T00140 C4O0QK 49821278 IC50 = 21 nM T00140 CI94KF 49864056 IC50 > 100000 nM T00140 CJG45C 49864057 IC50 > 100000 nM T00140 C4VWN3 49864058 IC50 > 100000 nM T00140 C3PX9L 49864059 IC50 > 100000 nM T00140 C63CNQ 49864060 IC50 > 100000 nM T00140 C8YC0P 49864071 IC50 = 22000 nM T00140 C2CNR6 49864072 IC50 = 49000 nM T00140 CKV94U 49864073 IC50 = 9000 nM T00140 CP2N7E 50925496 IC50 = 31 nM T00140 CX3NI6 50925497 IC50 = 28 nM T00140 C64KTI 51042131 IC50 = 7400 nM T00140 CHKL90 51042348 IC50 > 10000 nM T00140 CJA40Y 51109711 IC50 = 300 nM T00140 C4R8ZK 51136453 IC50 = 8100 nM T00140 CZD5R6 51346789 IC50 = 2300 nM T00140 C84JTI 51346790 IC50 = 260 nM T00140 C7SY9Q 51353746 IC50 = 2110 nM T00140 C3YZE7 51353747 IC50 = 580 nM T00140 C0Y1FD 51353749 IC50 = 320 nM T00140 CM8H9U 51353750 IC50 = 630 nM T00140 C86QEY 51353751 IC50 = 110 nM T00140 C9T0IK 51354048 IC50 = 130 nM T00140 CD75RU 51354049 IC50 = 120 nM T00140 CPG1R7 51354050 IC50 = 110 nM T00140 C4MH8K 51355427 IC50 = 6700 nM T00140 CNJ4A8 51355697 IC50 = 900 nM T00140 CWZ94B 51355698 IC50 = 27000 nM T00140 CM2SH9 51355699 IC50 > 30000 nM T00140 C6CEN7 51355700 IC50 = 9300 nM T00140 CG4L0N 51355701 IC50 > 30000 nM T00140 C6T1IN 51355702 IC50 > 30000 nM T00140 C0X3DU 51355965 IC50 = 8800 nM T00140 CEXJ19 51355966 IC50 > 30000 nM T00140 C2XGZ3 51355967 IC50 = 600 nM T00140 CYE47P 51355968 IC50 = 2800 nM T00140 CSK29T 51355969 IC50 > 30000 nM T00140 CS9V6B 51356246 IC50 = 1700 nM T00140 C04TKO 51356247 IC50 > 30000 nM T00140 CIT7W2 51534485 IC50 = 1600 nM T00140 C9YOV2 52102419 IC50 = 90 nM T00140 COK7Q1 52941460 IC50 > 20000 nM T00140 CVT1A7 52941563 IC50 = 154 nM T00140 C7N6RA 52941564 IC50 > 10000 nM T00140 C58DMR 53252516 IC50 > 50000 nM T00140 CP7Q0N 53316966 IC50 = 6000 nM T00140 C6JEY7 53317141 IC50 = 4400 nM T00140 C6G7ZT 53317142 IC50 = 700 nM T00140 CHN76K 53318433 IC50 = 170 nM T00140 CFP6I8 53319766 IC50 = 400 nM T00140 C89KRP 53321057 IC50 = 240 nM T00140 CQ06BD 53325026 IC50 = 600 nM T00140 CGS68Y 53325027 IC50 = 300 nM T00140 C4J5DH 53326328 IC50 = 500 nM T00140 C6JUK8 53326329 IC50 = 2000 nM T00140 CF1E3L 53358320 IC50 = 5500 nM T00140 CC7KT6 53363130 IC50 = 7200 nM T00140 CF5U2R 53363131 IC50 = 600 nM T00140 CSC3V7 53363132 IC50 = 4700 nM T00140 CH2DO7 53363133 IC50 = 700 nM T00140 CPD82G 53363134 IC50 = 2100 nM T00140 CI4D2P 53363220 IC50 = 6000 nM T00140 C2O8FZ 53363221 IC50 > 10000 nM T00140 CX7I2Y 53363222 IC50 = 900 nM T00140 C5H6YT 53363223 IC50 = 800 nM T00140 C1WB4D 53363224 IC50 = 900 nM T00140 CUI04W 53363313 IC50 = 300 nM T00140 CY3OX0 53363314 IC50 = 200 nM T00140 C8G0LH 53363315 IC50 = 400 nM T00140 CB34MJ 53363401 IC50 = 800 nM T00140 C7WAJ2 53439651 IC50 = 400 nM T00140 C1EFU6 53483951 IC50 > 50000 nM T00140 CM8W2Z 53766704 IC50 = 50 nM T00140 CQRS73 54580674 IC50 > 10000 nM T00140 CFE2A6 54581686 IC50 > 10000 nM T00140 C9LMW2 54583638 IC50 = 800 nM T00140 C6LTB2 54585561 IC50 > 10000 nM T00140 CB2C9S 54754352 IC50 = 2800 nM T00140 COL43S 54754353 IC50 = 2500 nM T00140 C5GRB6 54754354 IC50 = 2000 nM T00140 C3YM2E 54754518 IC50 = 1600 nM T00140 C43YCF 54878877 IC50 = 2237 nM T00140 CGC8D1 56598067 IC50 = 300 nM T00140 CXV96Y 56598068 IC50 = 150 nM T00140 CN3F5O 56641761 IC50 = 8000 nM T00140 C7ZI3H 56642018 IC50 > 10000 nM T00140 CV4YS2 56642150 IC50 = 2900 nM T00140 CZ6IY2 56642151 IC50 = 2900 nM T00140 CTM21L 56642287 IC50 = 2600 nM T00140 C6TVB8 56642288 IC50 = 8000 nM T00140 CV82SU 56642289 IC50 = 2900 nM T00140 CU1G5A 56642290 IC50 = 3500 nM T00140 CT50SH 56642418 IC50 = 2800 nM T00140 CG06ZW 56642419 IC50 = 3000 nM T00140 C5ICJ1 56642420 IC50 = 3300 nM T00140 CNL5G9 56642421 IC50 > 10000 nM T00140 CJ60HC 56642535 IC50 = 8000 nM T00140 C0SM7Z 56642536 IC50 = 4000 nM T00140 C6TLW3 56642537 IC50 > 10000 nM T00140 CG1N9O 56838295 IC50 = 100 nM T00140 CL16UQ 56949326 IC50 < 10000 nM T00140 C26UYE 56968384 IC50 > 100000 nM T00140 CY49QF 56968385 IC50 > 100000 nM T00140 CI2TP8 56968386 IC50 > 100000 nM T00140 CW25NO 56968387 IC50 = 69000 nM T00140 CBM48V 56968388 IC50 = 72000 nM T00140 CY8W7U 56968389 IC50 = 80000 nM T00140 C1YPA9 56968390 IC50 = 80000 nM T00140 CD87NY 56968391 IC50 = 41000 nM T00140 C6J1NL 56968615 IC50 = 62000 nM T00140 CMAG09 56968616 IC50 = 12000 nM T00140 CKI4A5 56968617 IC50 = 8000 nM T00140 CRF5N6 57390428 IC50 = 50 nM T00140 CI7X3V 57390429 IC50 = 30 nM T00140 CB1R8Z 57393138 IC50 = 270 nM T00140 CA72OL 57393840 IC50 = 25800 nM T00140 C7CN0I 57393841 IC50 = 13500 nM T00140 CS52FT 57393844 IC50 = 360 nM T00140 CAXT47 57393845 IC50 = 3090 nM T00140 CCP05K 57394873 IC50 = 1200 nM T00140 CAQ1V7 57395579 IC50 = 180 nM T00140 CML32C 57396634 IC50 = 1760 nM T00140 CN89AW 57396635 IC50 = 610 nM T00140 CU7O4B 57397391 IC50 = 3450 nM T00140 CR8YB4 57397392 IC50 = 6050 nM T00140 CW1K5I 57397393 IC50 = 91100 nM T00140 CYVE39 57397507 IC50 = 260 nM T00140 C0W1DF 57397555 IC50 = 80 nM T00140 C21RJC 57398407 IC50 = 150 nM T00140 CD3WE1 57398408 IC50 = 60 nM T00140 CICN26 57398409 IC50 = 60 nM T00140 CH94OE 57398410 IC50 = 500 nM T00140 C5QBK1 57400809 IC50 = 680 nM T00140 C7S4QK 57401877 IC50 = 420 nM T00140 CU6W9N 57402570 IC50 = 350 nM T00140 CFV7C6 57402705 IC50 = 430 nM T00140 CGO46T 57403590 IC50 = 6100 nM T00140 CVR24Z 58911052 IC50 = 400 nM T00140 C34XUR 60165328 IC50 = 116 nM T00140 CV0R6S 60168009 IC50 = 80 nM T00140 CWM6A0 60168044 IC50 = 8000 nM T00140 C9YE0M 60200527 IC50 = 6000 nM T00140 CLM07N 60200528 IC50 = 5000 nM T00140 C01PGH 60200529 IC50 = 5300 nM T00140 CHW2I8 66571763 IC50 = 6100 nM T00140 C5K2CY 66571764 IC50 > 10000 nM T00140 CY4X5D 66571765 IC50 > 10000 nM T00140 C0G1LM 66571766 IC50 > 10000 nM T00140 CKT32E 66571767 IC50 > 10000 nM T00140 C1P3RA 66571860 IC50 = 2000 nM T00140 CTW74V 66571861 IC50 > 10000 nM T00140 CES4Y3 66571862 IC50 = 6800 nM T00140 CF96OW 66571863 IC50 > 5000 nM T00140 C5H2ZY 66571963 IC50 = 900 nM T00140 C7YPV3 66571964 IC50 = 2000 nM T00140 CX04YA 66571965 IC50 = 1200 nM T00140 C8DY7B 66573411 IC50 > 10000 nM T00140 C0B7CK 66573412 IC50 > 10000 nM T00140 C5I3XH 66573413 IC50 > 10000 nM T00140 COAP48 67502417 IC50 = 6100 nM T00140 CL3RX8 67504002 IC50 = 2600 nM T00140 C9SMV3 68815772 IC50 = 9900 nM T00140 CE9KU0 70681522 IC50 = 210 nM T00140 C9T1MJ 70681523 IC50 = 100 nM T00140 C5LSD6 70681524 IC50 = 150 nM T00140 CDV38Z 70681525 IC50 = 760 nM T00140 C5GU9E 70681526 IC50 = 3550 nM T00140 C49YHM 70681528 IC50 = 140 nM T00140 CT4H7V 70681529 IC50 = 60 nM T00140 CBD54X 70683632 IC50 = 140 nM T00140 CE4R5H 70683633 IC50 = 80 nM T00140 CU7AX6 70683634 IC50 = 70 nM T00140 C21SAP 70683635 IC50 = 90 nM T00140 CTM0A8 70685770 IC50 = 200 nM T00140 C8C3ID 70685771 IC50 = 80 nM T00140 CFJY31 70685772 IC50 = 900 nM T00140 C3VU2Z 70687905 IC50 = 180 nM T00140 CL8AM3 70687906 IC50 = 260 nM T00140 CZL41X 70689933 IC50 = 80 nM T00140 C78WJZ 70689934 IC50 = 2140 nM T00140 C60MUF 70689935 IC50 = 130 nM T00140 CFH9V4 70692088 IC50 = 90 nM T00140 C04UAT 70692089 IC50 = 80 nM T00140 CI54AW 70692090 IC50 = 1990 nM T00140 CW3JB2 70694133 IC50 = 90 nM T00140 CI5U0X 70694134 IC50 = 130 nM T00140 CUF2K4 70695683 IC50 = 32 nM T00140 CE6RV8 70696266 IC50 = 210 nM T00140 C8VTG7 70696267 IC50 = 4660 nM T00140 CA76MQ 70701378 IC50 > 35000 nM T00140 CGWB74 70701426 IC50 > 100000 nM T00140 CT4IL7 70701432 IC50 > 100000 nM T00140 CI7Z8X 70701462 IC50 > 50000 nM T00140 CM34VK 70701465 IC50 > 50000 nM T00140 CE25CT 70701468 IC50 > 50000 nM T00140 C2COY0 71296422 IC50 = 600 nM T00140 CTZ59M 71307312 IC50 = 1670 nM T00140 CAQH38 71359348 IC50 > 50000 nM T00140 CKZ6W7 71394041 IC50 = 290 nM T00140 CS3RK5 71451782 IC50 = 2000 nM T00140 CUA81S 71451783 IC50 = 1500 nM T00140 C53HRS 71451785 IC50 = 2300 nM T00140 C7HVK4 71453597 IC50 = 3500 nM T00140 CV8N3Q 71453598 IC50 = 900 nM T00140 CWYG47 71455331 IC50 = 3700 nM T00140 CFJC03 71455332 IC50 = 3900 nM T00140 CB34ZQ 71455333 IC50 = 4700 nM T00140 CRS19Y 71457107 IC50 = 1700 nM T00140 CB1Q5R 71458972 IC50 = 5000 nM T00140 CL16CK 71458973 IC50 = 2500 nM T00140 CPVC31 71460125 IC50 > 50000 nM T00140 CH3YD6 71460772 IC50 = 1600 nM T00140 C9HK3Z 71462499 IC50 = 6800 nM T00140 CCDU47 71462500 IC50 = 2900 nM T00140 C0GJ4U 71493002 IC50 = 229 nM T00140 CWL1C8 71561507 IC50 = 600 nM T00140 CKV8A9 71561508 IC50 = 1000 nM T00140 C7R5EZ 71571581 IC50 = 400 nM T00140 CCZ3A4 71574951 IC50 = 1467 nM T00140 CT7I1M 71574952 IC50 = 1540 nM T00140 CR45LK 71575134 IC50 = 842 nM T00140 C9L4OE 71575135 IC50 = 439 nM T00140 C1J8ZR 71575136 IC50 = 191 nM T00140 C6XA4W 71575233 IC50 = 336 nM T00140 C8A5YG 71575234 IC50 = 696 nM T00140 C6XR5B 71575235 IC50 = 649 nM T00140 C47GVA 71575236 IC50 = 473 nM T00140 CK0W3S 71575346 IC50 = 614 nM T00140 CIK2H4 71575347 IC50 = 558 nM T00140 CPX09S 71575348 IC50 = 620 nM T00140 C6O7LP 71575349 IC50 = 459 nM T00140 C5CLE8 71575350 IC50 = 480 nM T00140 CC0D1M 71575458 IC50 = 439 nM T00140 CE0TN5 71575459 IC50 = 1107 nM T00140 C1XA7Z 71575460 IC50 = 1593 nM T00140 C61AXK 71575461 IC50 = 253 nM T00140 C5C3SP 71575560 IC50 = 192 nM T00140 CI7K0M 71575561 IC50 = 189 nM T00140 CQU1T8 71575562 IC50 = 190 nM T00140 CTZ65E 71718877 IC50 = 1000 nM T00140 CB25FU 71719484 IC50 = 1000 nM T00140 C2C6QY 71720724 IC50 = 5000 nM T00140 C6Z8PV 71725229 IC50 = 400 nM T00140 C8HZ6U 71764503 IC50 > 10000 nM T00140 CGF6Z3 72195591 IC50 > 10000 nM T00140 C6KIP1 72195592 IC50 = 4000 nM T00140 COBU91 72375187 IC50 = 6300 nM T00140 C74HXD 72375188 IC50 > 10000 nM T00140 C2OZ9H 72375189 IC50 = 6800 nM T00140 CUB64C 72546190 IC50 = 1800 nM T00140 COI3K8 72548264 IC50 = 23500 nM T00140 CPB90G 72548265 IC50 = 3400 nM T00140 C5QCN8 72715707 IC50 = 6500 nM T00140 C3D8VG 72715708 IC50 = 8700 nM T00140 CMFD46 72734874 IC50 = 800 nM T00140 C2K0GM 72734875 IC50 = 3800 nM T00140 CBO3D4 72734876 IC50 = 3600 nM T00140 CUH2V3 72734877 IC50 = 2900 nM T00140 CD82PY 72734878 IC50 > 10000 nM T00140 CZWL24 72734879 IC50 = 700 nM T00140 C6WKI3 72735052 IC50 = 2000 nM T00140 C3QIV9 72735053 IC50 = 200 nM T00140 CXZ2Q1 72735054 IC50 = 700 nM T00140 CPN87X 72735055 IC50 = 400 nM T00140 C4TLU8 72735056 IC50 = 200 nM T00140 CWHB65 72735057 IC50 = 1500 nM T00140 CG1PX4 72735224 Ki = 70300 nM T00140 CZB62X 72735237 IC50 = 1500 nM T00140 CU07KO 72735238 IC50 = 1400 nM T00140 CKH6N5 72735239 IC50 = 400 nM T00140 CQBP32 72735240 IC50 = 400 nM T00140 C9OXI7 72735241 IC50 = 600 nM T00140 C1DI9G 72735242 IC50 = 800 nM T00140 CWU6C4 72735414 IC50 = 300 nM T00140 CFNK27 72735415 IC50 = 1800 nM T00140 CB3SU5 72735416 IC50 = 5000 nM T00140 CF8N6W 72735417 IC50 = 600 nM T00140 CX2ND4 72735418 IC50 = 1600 nM T00140 CVX16U 72735589 IC50 = 700 nM T00140 CSDF35 72735590 IC50 = 600 nM T00140 C4JSP6 72735591 IC50 = 1900 nM T00140 CH5CF9 72735592 IC50 = 400 nM T00140 CG9JU0 72735593 IC50 = 900 nM T00140 CWJS67 72793857 IC50 = 1500 nM T00140 CPDL08 73052732 IC50 = 6700 nM T00140 C2RZ8J 73052890 IC50 = 1300 nM T00140 CTY72V 73052891 IC50 = 3200 nM T00140 CKR84E 73052892 IC50 = 730 nM T00140 CKC43H 73052893 IC50 = 460 nM T00140 C2B4OF 73053041 IC50 = 1200 nM T00140 C16YKH 73053042 IC50 = 1800 nM T00140 C5XO2M 73348950 IC50 = 700 nM T00140 C7INR4 73356550 IC50 = 500 nM T00140 C32DPL 76310435 Ki = 8.4 nM T00140 CBZ6O4 76310436 Ki = 2530 nM T00140 CRFO59 76310437 Ki = 95 nM T00140 CWQ31O 76314095 IC50 = 5460 nM T00140 CNV01E 76317665 IC50 = 8330 nM T00140 C7MR0A 76321372 IC50 = 14 nM T00140 CEM2R9 76324599 IC50 = 600 nM T00140 C5WTG1 76328546 IC50 = 3500 nM T00140 CPD8I6 76328547 IC50 = 8 nM T00140 CLDI40 76328548 IC50 = 2980 nM T00140 CH2WZ0 76331903 IC50 = 30 nM T00140 C8RZC0 76332104 IC50 = 280 nM T00140 C47ZQI 76332223 IC50 = 130 nM T00140 C0RVU2 76332224 Ki = 320 nM T00140 CIS0R8 76335724 IC50 = 2100 nM T00140 C94JNM 76335864 Ki = 9.9 nM T00140 C5CQW0 76335865 Ki = 510 nM T00140 CWJ4N9 77461129 IC50 = 850 nM T00140 C3O8NL 78427626 IC50 = 5700 nM T00140 CL3XS0 81689867 IC50 = 30 nM T00140 CU36EM 85998423 IC50 = 100 nM T00140 CFW5C9 90643727 IC50 = 9100 nM T00140 CE23GV 90643728 IC50 = 3800 nM T00140 C8BV9Q 90643729 IC50 = 3200 nM T00140 CC94JU 90643730 IC50 = 800 nM T00140 C8HM9U 90643731 IC50 = 800 nM T00140 CQA2B7 90643732 IC50 = 1800 nM T00140 C12JEM 90643733 IC50 = 230 nM T00140 CL6X2D 90643734 IC50 = 2300 nM T00140 COP83K 90643735 IC50 = 900 nM T00140 CN15BS 90643736 IC50 = 800 nM T00140 CJ61WQ 90643737 IC50 = 4200 nM T00140 C35WMJ 90643738 IC50 = 2900 nM T00140 CD1L4M 90643930 IC50 = 250 nM T00140 C1Z7VS 90643931 IC50 = 60 nM T00140 C9A6DF 90643932 IC50 = 700 nM T00140 C84YLF 90643933 IC50 > 50000 nM T00140 CD38OH 90643934 IC50 > 50000 nM T00140 C2TXO6 90643935 IC50 = 14900 nM T00140 CU6E0X 90644814 IC50 = 8100 nM T00140 C14PVH 90644815 IC50 = 80200 nM T00140 C9DI3W 90654808 IC50 = 30 nM T00140 C4SV2M 90654809 IC50 = 14400 nM T00140 C6KA5S 117872651 IC50 = 1600 nM T00140 C4QA9X 118536041 IC50 = 16300 nM T00140 CAG8I9 118536042 IC50 = 480 nM T00140 C6JPZ0 118536045 IC50 = 5900 nM T00140 CTV45Z 118536050 IC50 = 380 nM T00140 CO78DP 118536053 IC50 = 6100 nM T00140 C7HEO0 118536059 IC50 = 7400 nM T00140 COVA12 118536071 IC50 = 6000 nM T00140 CKRN05 118708820 IC50 = 4400 nM T00140 CX38JV 118708821 IC50 = 30 nM T00140 CC9Q1X 118708822 IC50 = 3300 nM T00140 C2CK0E 118708823 IC50 = 400 nM T00140 CJZW48 118708824 IC50 = 50 nM T00140 C6TFM1 118708825 IC50 = 600 nM T00140 CIRM37 118708871 IC50 > 10000 nM T00140 C0UT4S 118719671 IC50 = 580 nM T00140 CP8VO2 118719672 IC50 = 3610 nM T00140 C9MOL3 118719673 IC50 = 8360 nM T00140 C0GRV7 118719674 IC50 = 580 nM T00140 CBD8H2 118719675 IC50 = 250 nM T00140 CKJ41L 118719676 IC50 = 190 nM T00140 C5W8YD 118719677 IC50 = 1070 nM T00140 C92GWV 118719678 IC50 = 520 nM T00140 CR9KU8 118719679 IC50 = 1660 nM T00140 CUE76I 118719680 IC50 = 330 nM T00140 CR9W1Y 118719681 IC50 = 330 nM T00140 C7K1SP 118719682 IC50 = 280 nM T00140 CU7C6E 118719683 IC50 = 1580 nM T00140 CO3B8Q 118719685 IC50 = 6090 nM T00140 CX1EH8 118719686 IC50 = 6040 nM T00140 CZP7L8 118719687 IC50 = 960 nM T00140 C78KPR 118719688 IC50 = 440 nM T00140 C7FMG1 118719689 IC50 = 2870 nM T00140 C41FDZ 118719690 IC50 = 4620 nM T00140 CD23PM 118719692 IC50 = 10280 nM T00140 C6QFU3 118719693 IC50 = 1860 nM T00140 CF7P1Q 118719694 IC50 = 8220 nM T00140 CY0BA2 118719695 IC50 > 30000 nM T00140 C93GET 118719696 IC50 = 940 nM T00140 CCG49W 118719697 IC50 = 6150 nM T00140 CSF90I 118719698 IC50 = 350 nM T00140 CGJ6T0 118719699 IC50 = 120 nM T00140 CDB5C1 118719700 IC50 = 350 nM T00140 CF19PW 118719701 IC50 = 1560 nM T00140 C43AXD 118719702 IC50 = 200 nM T00140 CUK4Q2 118719703 IC50 = 430 nM T00140 CNZ0F7 118719704 IC50 = 1500 nM T00140 C0T3KI 118719705 IC50 = 10 nM T00140 C2CR5L 118719706 IC50 = 80 nM T00140 CBN35M 118719707 IC50 = 120 nM T00140 CTXA23 118726936 IC50 = 5700 nM T00140 C2FWY0 118726937 IC50 = 2100 nM T00140 C6XH0K 118726938 IC50 = 550 nM T00140 CE7L6H 118726939 IC50 = 750 nM T00140 CB23OM 118726943 IC50 = 500 nM T00140 CVU2B8 118726944 IC50 = 300 nM T00140 C7EU9N 118726945 IC50 = 300 nM T00140 CXEG20 118726946 IC50 = 2300 nM T00140 CMS2J7 118726947 IC50 = 700 nM T00140 CHM38G 118726948 IC50 = 900 nM T00140 CY3J0G 118726949 IC50 = 200 nM T00140 C94HSX 118726950 IC50 = 6700 nM T00140 CR6IC4 118726951 IC50 = 200 nM T00140 C4J5EW 118726952 IC50 = 900 nM T00140 CVO6Y5 118726954 IC50 = 250 nM T00140 CA8TS2 118726955 IC50 = 1700 nM T00140 C89LIX 118726956 IC50 = 500 nM T00140 CH56WO 118733904 IC50 = 2000 nM T00140 C13QDH 118733905 IC50 = 170 nM T00140 CHL8O4 118733906 IC50 = 190 nM T00140 CGA8F3 118733907 IC50 = 1800 nM T00140 CW8Y1Z 118733908 IC50 > 10000 nM T00140 CD29YZ 118733909 IC50 > 10000 nM T00140 CLVK83 118733910 IC50 = 3000 nM T00140 C83YDG 118733911 IC50 = 560 nM T00140 C2QZ3C 118733912 IC50 = 4100 nM T00140 C9K0BS 118733913 IC50 = 1900 nM T00140 CAZN10 118733914 IC50 = 3400 nM T00140 CH1KO7 118733915 IC50 = 2600 nM T00140 CQ78LB 118733916 IC50 = 320 nM T00140 CAP25H 118734013 IC50 = 490 nM T00140 C2P5US 118734014 IC50 = 450 nM T00140 CT6JH4 118734015 IC50 = 1700 nM T00140 CJ3N9V 118734016 IC50 = 990 nM T00140 CJ8E2Z 118734017 IC50 = 330 nM T00140 CW38MF 118734018 IC50 = 130 nM T00140 C8D6VE 118734019 IC50 = 60 nM T00140 CDAQ62 118734020 IC50 = 29 nM T00140 CQ4N1V 118734021 IC50 = 50 nM T00140 C82UZC 118734022 IC50 = 90 nM T00140 CD08VT 118734023 IC50 = 620 nM T00140 CR52OC 118734025 IC50 = 380 nM T00140 CS9QP0 118734026 IC50 = 300 nM T00140 C2Y0AN 118735510 IC50 = 1900 nM T00140 CFRJ40 118735511 IC50 > 10000 nM T00140 CC56FQ 118735512 IC50 > 10000 nM T00140 CSKB62 122178788 IC50 = 350 nM T00140 C64DUW 122186832 IC50 > 10000 nM T00140 CTD1Q4 122186833 IC50 = 460 nM T00140 C0RTQ5 122186834 IC50 = 970 nM T00140 C9W7SY 122186835 IC50 = 2700 nM T00140 CQBF95 122186836 IC50 = 1600 nM T00140 C7U5XI 122186837 IC50 = 1600 nM T00140 CMGL28 122186838 IC50 = 1300 nM T00140 C8Z5MV 122186839 IC50 = 2800 nM T00140 CXT1Y6 122186841 IC50 = 2700 nM T00140 C7C0JB 122186842 IC50 = 8600 nM T00140 CBH2L6 122186843 IC50 = 2900 nM T00140 C8Q6JM 122188662 IC50 = 1800 nM T00140 CMP37E 122188663 IC50 = 920 nM T00140 C0NGP8 122188664 IC50 = 470 nM T00140 C09ROJ 122188665 IC50 = 180 nM T00140 CS0ZY2 122188666 IC50 = 8230 nM T00140 C3MVH6 122188667 IC50 > 10000 nM T00140 C7CG6F 122188668 IC50 = 1300 nM T00140 CIZP43 122188669 IC50 = 7400 nM T00140 CK1AL2 122188670 IC50 = 6100 nM T00140 CD9FR4 122188671 IC50 = 3100 nM T00140 CQLG08 122188672 IC50 = 200 nM T00140 CDZW91 122188673 IC50 > 10000 nM T00140 C5Z8ID 122188674 IC50 > 10000 nM T00140 CPW16U 122188675 IC50 = 7600 nM T00140 CF5M0J 122188676 IC50 = 600 nM T00140 C6B7VZ 122188677 IC50 = 160 nM T00140 CC73OV 122188678 IC50 = 2600 nM T00140 CT1QR5 122212238 IC50 = 12400 nM T00140 CV9S1Z 127025829 IC50 > 10000 nM T00140 C8R7GU 127025830 IC50 > 10000 nM T00140 CX0FO4 127027015 IC50 = 1260 nM T00140 C9L5ZT 127027059 IC50 = 257 nM T00140 C5OU9X 127027060 IC50 = 182 nM T00140 C78XDC 127027061 IC50 = 255 nM T00140 C1C7WU 127027062 IC50 = 657 nM T00140 C8H0ED 127027063 IC50 = 237 nM T00140 C2CV9A 127027383 IC50 = 170 nM T00140 CXLR24 127027708 IC50 = 220 nM T00140 CRL1Q6 127027709 IC50 = 170 nM T00140 CJPM87 127027710 IC50 = 290 nM T00140 C84IUE 127027711 IC50 = 200 nM T00140 CD6RK8 127027712 IC50 = 1150 nM T00140 C3F1ID 127027713 IC50 > 10000 nM T00140 CN6S5Z 127032928 IC50 > 10000 nM T00140 C6HA7R 127049680 IC50 > 10000 nM T00140 CQ02ED 129834645 IC50 = 2460 nM T00140 C4N3LI 132564656 IC50 = 10000 nM T00140 CQ6ZR1 132603681 IC50 = 1100 nM T00140 C4HN2Y 134155900 IC50 = 22800 nM T00140 C4O2KF 134601764 IC50 = 1790 nM T00140 CIZE14 134813912 IC50 = 900 nM T00140 CCA43U 135411779 IC50 > 30000 nM T00140 CNKD13 135423790 IC50 = 3300 nM T00140 C48NWF 135423791 IC50 = 3100 nM T00140 CEVL69 135423792 IC50 = 5800 nM T00140 C8RUP4 135432996 IC50 = 600 nM T00140 CERL46 135443011 IC50 = 1950 nM T00140 CSB0M9 135494223 IC50 = 13 nM T00140 C3YRK0 135495764 IC50 > 30000 nM T00140 CCO3K7 135580426 IC50 = 2600 nM T00140 C9IH2B 135601507 IC50 = 1900 nM T00140 C6JF0E 135616214 IC50 < 1000 nM T00140 C12FNX 135637726 IC50 = 5880 nM T00140 CR8SN6 135703034 IC50 = 3000 nM T00140 CP3L5K 135799334 IC50 = 2900 nM T00140 C3N2FJ 135906278 IC50 > 10000 nM T00140 CRS1W8 135934760 IC50 = 860 nM T00140 CR75VS 135972423 IC50 = 190 nM T00140 COK59P 135972424 IC50 > 5000 nM T00140 CH4YE6 135987613 IC50 = 1000 nM T00140 CI63QS 136056624 IC50 > 50000 nM T00140 CP8Z5H 136088955 IC50 = 650 nM T00140 CW4J5O 136224196 IC50 = 8000 nM T00140 C94ZVL 136240270 IC50 = 6250 nM T00140 C1WOF5 136241419 IC50 = 5550 nM T00140 C3RW4K 136244259 IC50 = 790 nM T00140 CST9B8 136244569 IC50 = 1900 nM T00140 CB6PC8 136254208 IC50 = 570 nM T00140 CSK95Y 136504263 IC50 = 13 nM T00140 C2W9NU 136998792 IC50 = 1070 nM T00140 C4VZ1D 137631727 IC50 = 1460 nM T00140 CB5J7A 137632811 IC50 = 490 nM T00140 C2HES1 137634058 IC50 = 2400 nM T00140 CGB4Q3 137634225 IC50 = 150 nM T00140 CI6N9P 137642063 IC50 = 6300 nM T00140 CX1CA4 137643130 IC50 = 28 nM T00140 CEP7V3 137643442 IC50 = 200 nM T00140 CZ97FD 137643716 IC50 = 260 nM T00140 C3F7GH 137649890 IC50 = 3600 nM T00140 CTCY45 137649934 IC50 = 2500 nM T00140 CGS7R9 137650981 IC50 = 550 nM T00140 CVRE58 137651602 IC50 = 1080 nM T00140 C1BYH6 137652930 IC50 = 1840 nM T00140 CHI80F 137652936 IC50 = 5000 nM T00140 C4A3XH 137653836 IC50 = 120 nM T00140 CV4JW5 137654468 IC50 = 100 nM T00140 C4SFA1 137658121 IC50 = 90 nM T00140 CY5S9B 139590192 IC50 = 900 nM T00140 CWM7G2 145950344 IC50 = 14.4 ug.mL-1 T00140 C3A1GS 145955474 IC50 > 10000 nM T00140 CO8RY0 145978927 IC50 = 3400 nM T00140 CLG8B6 145979296 IC50 = 8400 nM T00140 C1R3DV 145979732 IC50 = 240 nM T00140 C2NUH7 145979828 IC50 = 5500 nM T00140 C1D9ZU 145979972 IC50 > 100000 nM T00140 C1KO3V 145980102 IC50 = 4000 nM T00140 CW1C0E 145980212 IC50 = 130 nM T00140 COYB38 145980268 IC50 = 298 nM T00140 CC36AS 145980298 IC50 = 860 nM T00140 CW93VH 145980588 IC50 = 4200 nM T00140 C7QGD6 145980641 IC50 = 2760 nM T00140 CMRJ31 145980727 IC50 = 3500 nM T00140 C5OSG9 145980817 IC50 = 160 nM T00140 CM73GH 145981036 IC50 = 1300 nM T00140 C9XG2N 145981314 IC50 = 97500 nM T00140 CO84KR 145981339 IC50 = 110 nM T00140 CM02LY 145981376 IC50 = 500 nM T00140 C8TP1V 145981823 IC50 > 100000 nM T00140 CT31BN 145981863 IC50 = 2030 nM T00140 C3EDP1 145982139 IC50 = 2600 nM T00140 CHDB09 145982182 IC50 = 54300 nM T00140 CZQY07 145982329 IC50 = 500 nM T00140 CH3GA6 145982419 IC50 = 120 nM T00140 CFNJ87 145982457 IC50 = 9800 nM T00140 C1IBC7 145983185 IC50 = 700 nM T00140 CU95NM 145983649 IC50 = 600 nM T00140 CW4X2T 145984359 IC50 = 95100 nM T00140 C76ACJ 145985137 IC50 = 60 nM T00140 CM62SF 145985303 IC50 = 3200 nM T00140 CQ0F4H 145986097 IC50 = 300 nM T00140 CH1TE6 145986374 IC50 = 4400 nM T00140 CKO9H0 145986691 IC50 = 370 nM T00140 C5VJ0U 145986782 IC50 = 2100 nM T00140 C5V4BG 145986923 IC50 = 45 nM T00140 CQ7UX8 145986960 IC50 = 780 nM T00140 CVA7K0 145986989 IC50 = 860 nM T00140 C9M3YE 145987054 IC50 = 1360 nM T00140 C4ZBC9 145987188 IC50 = 3200 nM T00140 C1Y2VN 145987225 IC50 = 370 nM T00140 CG2J7C 145987315 IC50 = 1000 nM T00140 C21BYI 145987407 IC50 = 28900 nM T00140 C20LTV 145987586 IC50 = 130 nM T00140 CU03MH 145987714 IC50 = 300 nM T00140 C98DHT 145987800 IC50 > 100000 nM T00140 CA82TF 145987838 IC50 = 82400 nM T00140 C0WEB7 145987883 IC50 = 1400 nM T00140 C0RC3X 145988011 IC50 = 460 nM T00140 C3M1ZO 145988042 IC50 > 100000 nM T00140 C7DWP8 145988191 IC50 = 120 nM T00140 CE15SN 145988338 IC50 = 110 nM T00140 CI3V2U 145988600 IC50 = 1860 nM T00140 C10NDO 145988652 IC50 = 160 nM T00140 C1XU7P 145988798 IC50 > 100000 nM T00140 CFV79W 145989238 IC50 = 1240 nM T00140 C8SVA1 145989549 IC50 = 3300 nM T00140 CU1ET5 145990280 IC50 = 800 nM T00140 CM8K2G 145990428 IC50 = 94 nM T00140 CS38MY 145990546 IC50 = 782 nM T00140 C4JLA2 145990560 IC50 = 3790 nM T00140 C6RML9 145990587 IC50 = 100 nM T00140 CR59TZ 145990611 IC50 > 100000 nM T00140 C5QZJ4 145990784 IC50 = 15100 nM T00140 C3DE6F 145990898 IC50 = 370 nM T00140 CA69OZ 145991533 IC50 = 3200 nM T00140 CJ23ZQ 145991963 IC50 = 190 nM T00140 C14RPI 145992031 IC50 = 1100 nM T00140 CB9P8D 145992212 IC50 = 77600 nM T00140 CI45QF 145992217 IC50 = 4800 nM T00140 CBPF85 145992428 IC50 = 1060 nM T00140 CQ39BP 145992502 IC50 = 1700 nM T00140 C1WI3A 145992723 IC50 = 74300 nM T00140 C38CIQ 145992873 IC50 = 130 nM T00140 CF36AC 145993120 IC50 > 100000 nM T00140 C5YMR4 145993208 IC50 > 100000 nM T00140 C7QZ9D 145993245 IC50 = 1100 nM T00140 CQL0D9 145993288 IC50 = 900 nM T00140 CN8G1X 145993375 IC50 = 400 nM T00140 CUVC73 145993378 IC50 > 100000 nM T00140 C30CMY 145993498 IC50 > 100000 nM T00140 C27FDC 145993580 IC50 > 100000 nM T00140 CU80CE 145993587 IC50 = 1500 nM T00140 C2JHG5 145993960 IC50 = 6200 nM T00140 CNUM28 145994201 IC50 = 2400 nM T00140 C1VZ5D 155513018 IC50 = 9300 nM T00140 CO0GN6 155514213 IC50 > 10000 nM T00140 C2N6WF 155517734 IC50 > 10000 nM T00140 CQI2V8 155518055 IC50 = 560 nM T00140 C5B2IR 155518737 IC50 = 830 nM T00140 CJN65T 155519575 IC50 = 1010 nM T00140 C6VFM3 155521055 IC50 = 540 nM T00140 CA0T6X 155523257 IC50 = 240 nM T00140 CQKZ59 155523833 IC50 = 800 nM T00140 C3MW0Q 155523976 IC50 = 1100 nM T00140 C7BC2H 155525137 IC50 = 90 nM T00140 CG42OB 155528473 IC50 = 170 nM T00140 CL1ZG5 155530203 IC50 = 2200 nM T00140 C24KXE 155530411 IC50 = 80 nM T00140 CTEF18 155530430 IC50 = 70 nM T00140 CIJ3G0 155531569 IC50 = 2100 nM T00140 C5C7PV 155532437 IC50 = 2070 nM T00140 C2UW0O 155532784 IC50 = 2170 nM T00140 CH65JO 155533037 IC50 = 680 nM T00140 CZUC84 155534190 IC50 = 3000 nM T00140 CTH8F2 155534569 IC50 = 170 nM T00140 C76NZI 155535091 IC50 = 21000 nM T00140 C4P1XN 155536830 IC50 > 10000 nM T00140 C3S7VL 155537100 IC50 > 10000 nM T00140 CI3V4U 155537759 IC50 = 140 nM T00140 CCU6X3 155538568 IC50 = 10000 nM T00140 CAVL53 155539161 IC50 = 570 nM T00140 C3M6OK 155539896 IC50 = 900 nM T00140 C6C7AG 155539906 IC50 = 2300 nM T00140 CR9S6O 155542667 IC50 = 360 nM T00140 CA0WI7 155542837 IC50 = 5600 nM T00140 C9O4IW 155544859 IC50 = 640 nM T00140 CK5H3F 155545531 IC50 = 730 nM T00140 C9GFC0 155552295 IC50 > 10000 nM T00140 CUH67J 155556436 IC50 = 800 nM T00140 C3QT0N 155558153 IC50 = 720 nM T00140 CHGW35 155559094 IC50 = 1500 nM T00140 CT2X3Z 155560377 IC50 = 80 nM T00140 CT7PH4 155560482 IC50 = 120 nM T00140 C62UMN 155562130 IC50 = 890 nM T00140 CSB69O 155562385 IC50 = 570 nM T00140 CNL75J 155563178 IC50 = 900 nM T00140 C72LZA 155564090 IC50 = 1130 nM T00140 CO0KU6 155565005 IC50 = 10760 nM T00140 COKI17 155565163 IC50 = 530 nM T00140 CGZ14A 155566111 IC50 = 2090 nM T00140 COK1W3 155567033 IC50 = 420 nM T00140 CBK58I 155567041 IC50 = 2200 nM T00140 C40XPW 155567716 IC50 = 24000 nM T00140 D00AII 5281727 IC50 = 530 nM T00140 D00GBX 71751 IC50 = 4800 nM T00140 D00OTC 5385086 IC50 = 5480 nM T00140 D00YNY 753704 IC50 = 30 nM T00140 D01BZE 73659 IC50 > 40000 nM T00140 D01GSW 135433966 IC50 = 40 nM T00140 D01JYF 325144 IC50 = 15000 nM T00140 D01OFH 155160 IC50 = 1500 nM T00140 D01PBO 44423052 IC50 = 9200 nM T00140 D01SQY 128480 IC50 = 240 nM T00140 D02XEX 11168203 IC50 = 2700 nM T00140 D04DQJ 72303 IC50 = 4200 nM T00140 D05FJM 460087 IC50 = 4600 nM T00140 D05FKT 9960281 IC50 = 22 nM T00140 D05IQL 44158012 IC50 = 3400 nM T00140 D05MIV 5162 IC50 > 5000 nM T00140 D05PHI 14425906 IC50 = 2400 nM T00140 D05QOR 5280460 IC50 > 100000 nM T00140 D06DCK 44410706 IC50 = 2.3 nM T00140 D06OAH 448949 IC50 = 5700 nM T00140 D06TXM 24816385 IC50 = 2000 nM T00140 D06YGF 5281787 IC50 = 970 nM T00140 D06ZRX 5281717 IC50 = 18490 nM T00140 D07ARK 157806 IC50 = 150 nM T00140 D07CJR 5280733 IC50 = 2000 nM T00140 D07EAJ 10110469 IC50 = 450 nM T00140 D07EGB 3610 IC50 = 2800 nM T00140 D07JRW 10179787 IC50 = 14000 nM T00140 D07LUJ 64945 IC50 > 40000 nM T00140 D07TWV 123080 IC50 = 9500 nM T00140 D08IRN 18771543 IC50 = 350 nM T00140 D09OWE 92802 IC50 = 42000 nM T00140 D09VYW 9847548 IC50 = 3000 nM T00140 D0E0RW 69894 IC50 > 100000 nM T00140 D0F4HT 164272 IC50 = 100 nM T00140 D0F8QJ 5281813 IC50 = 2500 nM T00140 D0F9FG 46907602 IC50 = 18000 nM T00140 D0F9RO 6918774 IC50 > 40000 nM T00140 D0G3TK 5280863 IC50 = 2700 nM T00140 D0I9AT 73549 IC50 = 150 nM T00140 D0IO0I 6474893 IC50 = 5200 nM T00140 D0K7XQ 10561814 IC50 = 2500 nM T00140 D0LC7K 119034 IC50 > 40000 nM T00140 D0M6UM 129265 IC50 = 770 nM T00140 D0N7XM 24992964 IC50 = 5900 nM T00140 D0O0VZ 667639 IC50 = 240 nM T00140 D0O9NE 5388063 IC50 = 3620 nM T00140 D0PJ3M 637511 IC50 = 35000 nM T00140 D0Q9TL 44329500 IC50 = 190 nM T00140 D0R6ZC 9900113 IC50 = 1700 nM T00140 D0S0OE 5280383 IC50 = 2000 nM T00140 D0S0SH 10069117 IC50 = 107 nM T00140 D0S7ZQ 45267389 IC50 = 1400 nM T00140 D0SS4S 44158013 IC50 = 6900 nM T00140 D0U2YL 131820 IC50 = 37 nM T00140 D0U8IF 10114 IC50 = 24800 nM T00140 D0UH6R 44583183 IC50 = 38 nM T00140 D0V9EN 689043 IC50 = 8500 nM T00140 D0VC0I 5169 IC50 = 50 nM T00140 D0W3ZN 4712 IC50 = 50 nM T00140 D0Y0ES 3707 IC50 = 15000 nM T00140 D0Y1TA 45269978 IC50 = 4500 nM T00140 D0YJ3Q 5322065 IC50 = 2000 nM T42392 D00ENY 33032 Ki = 940 nM T42392 D03CNS 2910 EC50 = 2240 nM T42392 D02VKC 3272524 Ki = 210 nM T42392 D0B0NQ 127894 Ki = 2210 nM T42392 D04XMJ 11249042 Ki > 100000 nM T42392 D0A9VO 3538 Ki = 4000 nM T42392 D0M7MW 126758 EC50 = 100000 nM T42392 COC91V 10255 EC50 = 10570 nM T42392 C6T4AH 167842 Ki = 101 nM T42392 CC0E1V 447081 Ki = 3.89 nM T42392 CM41VL 656707 EC50 = 520 nM T42392 CMOR75 945544 EC50 = 25118.86 nM T42392 CZ6C2S 1316629 EC50 > 19952.62 nM T42392 C1EP3D 2733518 Ki = 250 nM T42392 CWK7X4 4694356 Ki = 370 nM T42392 CZU2N7 4862343 EC50 = 10000 nM T42392 C5H2IW 4862344 EC50 > 100000 nM T42392 C5Z8VG 6324635 Ki > 10000 nM T42392 CVW4L3 9795654 Ki = 19.3 nM T42392 C4CQ5B 9843690 EC50 = 398.11 nM T42392 C9TLQ4 9861035 Ki > 10000 nM T42392 CFV03Y 9926589 Ki = 117000 nM T42392 CFC2P8 9928016 EC50 = 150 nM T42392 CZ30AU 10013456 EC50 = 50582.47 nM T42392 C7Q1MJ 10132082 IC50 > 100000 nM T42392 CRJ2T0 10219992 Ki = 3680 nM T42392 C5PD0H 10330442 Ki = 3700 nM T42392 CFKJ76 10352480 Ki = 273 nM T42392 C9RO2X 10375113 Ki = 494 nM T42392 C7GIJ3 10398361 Ki = 280900 nM T42392 C1N2VM 10420002 Ki = 234 nM T42392 CXE7F5 10541731 Ki > 10000 nM T42392 C0O6ZI 10658567 EC50 > 3000000 nM T42392 CJZ04V 11096831 Ki = 115 nM T42392 CW0LO5 11121532 EC50 = 520 nM T42392 CR5XS2 11153198 Ki = 8260 nM T42392 CRS35K 11154806 Ki > 100000 nM T42392 CWB19Y 11161396 EC50 = 20400 nM T42392 CQ97KS 11198294 EC50 = 103 nM T42392 CA83CR 11199813 Ki = 5510 nM T42392 CQ38WM 11219775 Ki = 1610 nM T42392 CGRT02 11288627 Ki = 80.2 nM T42392 C2EA6X 11291212 EC50 = 73 nM T42392 CUTV05 11334126 IC50 = 1000 nM T42392 COD9Z2 11504477 EC50 = 5000 nM T42392 CH75CA 11508844 EC50 = 3200 nM T42392 C0SN2O 11515728 EC50 = 31622.78 nM T42392 CVO7T9 11522969 EC50 = 63095.73 nM T42392 CR83WI 11525569 EC50 = 1600 nM T42392 C29LCK 11537876 EC50 = 20000 nM T42392 C3VP9T 11544537 EC50 = 5011.87 nM T42392 C8V4UC 11544633 IC50 > 100000 nM T42392 CQ2X1J 11552469 EC50 = 6309.57 nM T42392 C84NIF 11566130 EC50 = 3162.28 nM T42392 CDFU34 11566489 EC50 = 7943.28 nM T42392 CJ3FH6 11568363 EC50 = 4000 nM T42392 CK96VD 11573153 Ki = 21000 nM T42392 C4IX6W 11573549 EC50 = 6309.57 nM T42392 C4AU8J 11574298 EC50 = 19952.62 nM T42392 CVX6K7 11580514 EC50 = 15848.93 nM T42392 CN1I8D 11581636 EC50 = 2500 nM T42392 CG24BP 11587814 EC50 = 10000 nM T42392 C1A3PZ 11595635 EC50 = 4000 nM T42392 CO1U3M 11610515 EC50 = 2500 nM T42392 C63MHR 11611549 EC50 = 2511.89 nM T42392 COW93C 11611844 EC50 = 5000 nM T42392 CB4G6F 11617056 EC50 > 50118.72 nM T42392 CB9MU1 11618681 EC50 = 7943.28 nM T42392 CPV49C 11632254 EC50 = 5000 nM T42392 C1R2BZ 11633045 EC50 = 4000 nM T42392 CCP69D 11638499 EC50 = 19952.62 nM T42392 CRT09O 11638500 EC50 = 19952.62 nM T42392 CPO25R 11647576 EC50 = 79400 nM T42392 CN6Y7D 11661294 EC50 = 6300 nM T42392 CE9W7N 11668999 EC50 = 1258.93 nM T42392 C6GVU2 11676790 EC50 = 300 nM T42392 C6TZ8Y 11683045 EC50 = 12589.25 nM T42392 CI6JR2 11684405 EC50 = 6300 nM T42392 CW4U3H 11688520 EC50 = 3162.28 nM T42392 CUDX43 11689005 EC50 > 50118.72 nM T42392 C6S2GN 11689802 EC50 = 7900 nM T42392 C8QIH0 11696657 EC50 = 5000 nM T42392 CQE1T6 11704038 EC50 > 50118.72 nM T42392 CL4DS1 11709762 EC50 = 15848.93 nM T42392 CIUV17 11711973 EC50 = 6200 nM T42392 CM1GA4 11773296 EC50 = 32 nM T42392 CHUX80 11818375 Ki = 2930 nM T42392 CDGZ79 11820131 Ki = 44900 nM T42392 CIO92V 16025391 EC50 = 23700 nM T42392 C3F4KH 16046205 EC50 = 97 nM T42392 CX2VU6 16046206 EC50 = 47 nM T42392 CQ2YP8 16659202 EC50 > 3000000 nM T42392 CS90PN 16718565 EC50 = 300 nM T42392 CZ3S6X 16732327 EC50 = 176300 nM T42392 C9PKX2 17747017 EC50 < 200000 nM T42392 CDZ2E6 18713992 EC50 = 150 nM T42392 CFAH74 20938953 EC50 = 2000 nM T42392 C6ORA8 24783140 EC50 > 19952.62 nM T42392 CN4Z2J 24825807 EC50 = 63095.73 nM T42392 C2S5PO 24825811 EC50 = 1995.26 nM T42392 C2MA5J 24825905 EC50 = 1000 nM T42392 C3YSN6 24826093 EC50 = 7943.28 nM T42392 C3LJ5E 24826094 EC50 = 31622.78 nM T42392 C7ZQ1U 24826095 EC50 = 19952.62 nM T42392 C46NAW 24826096 EC50 = 19952.62 nM T42392 C7Z1KI 24826368 EC50 = 10000 nM T42392 CSUI87 24826369 EC50 = 10000 nM T42392 CJ6Z9E 24826945 EC50 = 15848.93 nM T42392 CA29CU 24826946 EC50 = 39810.72 nM T42392 CY6QD7 24826947 EC50 = 31622.78 nM T42392 C1P3IL 24826949 EC50 = 31622.78 nM T42392 CM2Y0L 24827043 EC50 = 3981.07 nM T42392 CLM16X 24827044 EC50 = 1995.26 nM T42392 C2IB1S 24827045 EC50 = 3162.28 nM T42392 CHS35U 24827139 EC50 = 25118.86 nM T42392 C6OJ5C 24827142 EC50 = 31622.78 nM T42392 CL1K4P 24882540 Ki = 4000 nM T42392 C97QIV 24936160 EC50 < 300000 nM T42392 CI7NG8 24951587 EC50 = 10000 nM T42392 CEGV39 24951942 EC50 = 100000 nM T42392 C9EH3S 24951943 EC50 = 5011.87 nM T42392 CW9UN1 24951944 EC50 = 39810.72 nM T42392 CP98YL 24951946 EC50 = 19952.62 nM T42392 CVHP97 24951947 EC50 < 300000 nM T42392 C0UMZ2 24953726 EC50 = 10000 nM T42392 C8QD7Y 24967421 EC50 = 398.11 nM T42392 CA3D2O 24967783 EC50 = 794.33 nM T42392 CF0A5P 24984572 EC50 > 31622.78 nM T42392 C4E9IK 25015611 EC50 = 1000 nM T42392 CCE8S3 25015613 EC50 = 1258.93 nM T42392 C4U7OS 44152410 Ki = 53.1 nM T42392 CW9TR7 44346780 Ki = 16.7 nM T42392 C64ELF 44346789 Ki = 372 nM T42392 CQJW06 44346790 Ki = 461 nM T42392 C15MPO 44346798 Ki = 101 nM T42392 COQ86N 44416680 EC50 = 333 nM T42392 C84BWG 44416681 EC50 = 176 nM T42392 CBW5D3 44416682 EC50 = 1137 nM T42392 CAYR16 44416702 EC50 = 78 nM T42392 CXN16F 44416703 EC50 > 3000 nM T42392 C60GWQ 44416732 EC50 = 663 nM T42392 C1YW8F 44416748 EC50 = 174 nM T42392 CHD28J 44416750 EC50 > 3000 nM T42392 CQD2Y3 44416776 EC50 = 412 nM T42392 CIQ92O 44416794 EC50 = 965 nM T42392 C2YR8D 44416795 EC50 = 270 nM T42392 CIRK69 44416811 EC50 = 370 nM T42392 CCZW78 44416812 EC50 = 391 nM T42392 CE2NL6 44416834 EC50 = 280 nM T42392 C7PW9S 44416873 EC50 = 370 nM T42392 CAGW51 44416888 EC50 > 3000 nM T42392 C3ZIJ2 44416889 EC50 > 3000 nM T42392 CGH79E 44416892 EC50 = 395 nM T42392 CIW5X0 44416905 EC50 > 3000 nM T42392 CRB28F 44416986 EC50 = 36 nM T42392 CD3G7X 44417019 EC50 = 345 nM T42392 CD7JY5 44417039 EC50 = 426 nM T42392 CJS5Z7 44417040 EC50 = 111 nM T42392 CP71ZU 44417062 EC50 = 142 nM T42392 CPNL12 44417063 EC50 = 186 nM T42392 CYQ4C9 44417081 EC50 = 308 nM T42392 CK8FI3 44417082 EC50 = 42 nM T42392 CUKV64 44452462 Ki = 94000 nM T42392 C1TDN0 44555548 EC50 = 398.11 nM T42392 CL06SF 44555553 EC50 = 1000 nM T42392 CA8H6I 44555607 EC50 = 2511.89 nM T42392 CZ08MS 44555610 EC50 = 2511.89 nM T42392 CI57SU 44555667 EC50 = 100 nM T42392 CN90JW 44555668 EC50 = 1258.93 nM T42392 CPK75R 44555669 EC50 = 1258.93 nM T42392 C3PW2U 44555670 EC50 = 794.33 nM T42392 C0IAU9 44555671 EC50 = 1258.93 nM T42392 C31GAN 44555728 EC50 = 1000 nM T42392 CMX53V 44555729 EC50 = 3981.07 nM T42392 CIA98N 44555730 EC50 = 158.49 nM T42392 CQ13JF 44555733 EC50 = 100 nM T42392 C8KBI7 44556365 EC50 = 398.11 nM T42392 CI70YG 44556366 EC50 = 501.19 nM T42392 C9MX5Y 44608185 EC50 = 48200 nM T42392 C2L4HR 46238075 EC50 = 489000 nM T42392 CJB07Z 46238077 EC50 = 489778.82 nM T42392 CQX93F 46398805 EC50 = 2500 nM T42392 CO8RI0 46900136 EC50 = 794.33 nM T42392 CWR9M5 46900138 EC50 = 1995.26 nM T42392 CGN7Q8 46900139 EC50 = 1995.26 nM T42392 C5XJS2 49863866 EC50 = 398.11 nM T42392 C07DIE 49870853 EC50 = 100 nM T42392 CW6LP3 50992864 EC50 = 19952.62 nM T42392 C6UN8M 50992932 EC50 = 2511.89 nM T42392 CZ6NO1 50992933 EC50 = 1258.93 nM T42392 C38AOG 51087450 EC50 = 830 nM T42392 C1FX6A 52941684 EC50 = 400 nM T42392 CN9O7H 52941909 EC50 < 300000 nM T42392 CHV52T 52943128 EC50 < 300000 nM T42392 CVZ13N 52945564 EC50 = 1600 nM T42392 CUWT60 52945897 EC50 = 1980000 nM T42392 CK5VU2 52946383 EC50 = 300 nM T42392 CEU2N1 52947551 EC50 = 500 nM T42392 CGCK63 52947618 EC50 = 300 nM T42392 CDN06O 52948827 EC50 = 300 nM T42392 CM20WN 52949797 EC50 = 20000 nM T42392 CYQT21 53259006 EC50 = 710 nM T42392 COM3X0 53304137 EC50 = 46.13 nM T42392 C68CTA 53304138 EC50 = 3190 nM T42392 C5OGL3 53304139 EC50 = 1.995 nM T42392 C6YSX0 53304140 EC50 = 1819.7 nM T42392 CI2L3C 53304141 EC50 = 450 nM T42392 C2GIX4 53318967 EC50 > 31622.78 nM T42392 CN3X5S 53319053 EC50 = 1995.26 nM T42392 CPI8E5 53321322 EC50 = 501.19 nM T42392 CX6Z3Y 53323974 EC50 = 1258.93 nM T42392 C6OM2V 53323975 EC50 = 7943.28 nM T42392 CN8O2M 53325272 EC50 = 1584.89 nM T42392 C5DO3F 53325273 EC50 = 5011.87 nM T42392 CE53JT 53326549 EC50 = 1258.93 nM T42392 CRP3A6 56593692 Ki = 3150 nM T42392 CDT01W 60023862 Ki = 6400 nM T42392 CK7H6W 60023863 Ki = 128000 nM T42392 C86SPH 60023864 Ki = 238000 nM T42392 CJL45I 60023870 Ki = 3500 nM T42392 C0OFZ7 60023874 Ki = 77000 nM T42392 CB5X4L 60023875 Ki = 6200 nM T42392 CWV2O7 67530213 EC50 = 9060 nM T42392 C4G8FM 67531324 EC50 = 810 nM T42392 CD54OC 68586104 Ki = 22000 nM T42392 C5U0FY 68586486 Ki = 42000 nM T42392 CQ2XT7 68588179 Ki = 8800 nM T42392 CZ6UN9 68588451 Ki = 151000 nM T42392 C7SBU2 68590056 Ki = 19000 nM T42392 C9P7GB 69508277 EC50 = 7620 nM T42392 CDNJ51 69972507 Ki = 553000 nM T42392 CZH05N 71719873 Ki = 560000 nM T42392 CT3GH6 72543949 Ki = 30000 nM T42392 CY67ZT 72543950 Ki = 252000 nM T42392 C10GMK 72544188 Ki = 181000 nM T42392 CMG1J3 72544190 Ki = 2700 nM T42392 C7S2RQ 72544191 Ki = 400 nM T42392 C76VSM 72544192 Ki = 12000 nM T42392 CQ90OK 72544193 Ki = 5200 nM T42392 CT30EV 72544414 Ki = 2000 nM T42392 C92PSD 72544415 Ki = 2300 nM T42392 CYO4F3 72544417 Ki = 450000 nM T42392 C1HK0F 72544419 Ki = 13000 nM T42392 C0ARY4 72544635 Ki = 1700 nM T42392 C3F0SH 72544637 Ki = 3 nM T42392 C2KTJ7 72544639 Ki = 2200 nM T42392 CRI79J 72544641 Ki = 4400 nM T42392 C91VEK 72544642 Ki = 20000 nM T42392 CHM5L1 72544859 Ki = 12000 nM T42392 CRT02N 72544861 Ki = 335000 nM T42392 CD14GW 72544863 Ki = 17000 nM T42392 C3W2SA 72544865 Ki = 9600 nM T42392 C3EBZ6 72544866 Ki = 9600 nM T42392 CXG0P9 72546282 Ki = 1420000 nM T42392 CE6ST8 72546283 Ki = 15000 nM T42392 C3B8TH 72546523 Ki = 9000 nM T42392 C3Z1PE 72546524 Ki = 418000 nM T42392 CXWI86 72546765 Ki = 3300 nM T42392 CUJ9A3 72547031 Ki = 70000 nM T42392 C2BEW8 72547032 Ki = 44000 nM T42392 CCO6B5 72547033 Ki = 913000 nM T42392 CZB27J 72547288 Ki = 93000 nM T42392 CVKD75 72547289 Ki = 107000 nM T42392 CBH2X5 72547290 Ki = 87000 nM T42392 CA21EV 72547291 Ki = 172000 nM T42392 CKNW59 72547534 Ki = 89000 nM T42392 CWSJ60 72547535 Ki = 111000 nM T42392 C1DTV4 72547536 Ki = 1470000 nM T42392 C6JZ4H 72547537 Ki = 818000 nM T42392 CVID16 73348020 Ki = 29600000 nM T42392 CG5PL8 73349560 Ki = 149000 nM T42392 CA2R1Y 76309877 Ki = 13000 nM T42392 CV52YL 76309878 Ki = 22000 nM T42392 C8VC7N 102515534 Ki = 2260 nM T42392 CJ2ER5 102515535 Ki = 84000 nM T42392 C7SY0E 118009185 EC50 = 13000 nM T42392 CM4CT8 118009256 EC50 = 1500 nM T42392 CK64SO 118009262 EC50 = 2300 nM T42392 CS69AR 118009384 EC50 = 34400 nM T42392 CQW61N 118009417 EC50 = 572 nM T42392 CRS0L6 118009479 EC50 = 28300 nM T42392 CSHJ98 118009524 EC50 = 60200 nM T42392 CV5O1S 118009526 EC50 = 1900 nM T42392 C3K2WB 118009634 EC50 = 972 nM T42392 CZ34OF 118009669 EC50 = 5500 nM T42392 C07WHN 118010095 EC50 = 10700 nM T42392 CSA0C3 118010141 EC50 = 204 nM T42392 C04MZF 118010226 EC50 = 4500 nM T42392 C14YIX 118010387 EC50 = 2400 nM T42392 CL61DS 118010607 EC50 = 8600 nM T42392 CASX13 118011037 EC50 = 9400 nM T42392 C1K6IC 118017591 EC50 = 245 nM T42392 CBE91G 118017599 EC50 = 1100 nM T42392 C69XGV 118017702 EC50 = 9800 nM T42392 C40GYH 118017736 EC50 = 32900 nM T42392 CCH7L0 118017739 EC50 = 37000 nM T42392 C87TKV 118017811 EC50 = 1200 nM T42392 CVY1C6 118017915 EC50 = 66200 nM T42392 CV6PS1 122438413 EC50 = 9100 nM T42392 C9Q6PB 122438535 EC50 = 6400 nM T42392 CWK35R 122630616 EC50 = 16000 nM T42392 C79ZCY 122630795 EC50 = 45000 nM T42392 C56NLW 127039193 EC50 > 1000000 nM T42392 C7ACT6 127045913 EC50 = 48 nM T42392 CJ5K2C 127045914 EC50 = 2500 nM T42392 C5B0WF 127045915 EC50 = 73 nM T42392 CXV89R 127046129 EC50 = 5500 nM T42392 C9J0SK 127046302 EC50 = 48700 nM T42392 CQT2V5 127046683 EC50 = 359 nM T42392 CQC9U4 134137374 EC50 = 410 nM T42392 C5URK7 134146341 EC50 = 2200 nM T42392 C9S4DO 134152062 EC50 = 210 nM T42392 C0A2OR 134153491 EC50 = 1300 nM T42392 CAV7G1 134153879 EC50 = 460 nM T42392 C3XJZ6 134157459 EC50 = 31000 nM T42392 CLH0O3 134828072 EC50 = 13.4 nM T42392 CYC4H5 135453303 IC50 = 7600 nM T42392 C3K7QV 137628313 EC50 = 1.259 nM T42392 C4UN2I 137635645 EC50 = 370 nM T42392 CJ0GU7 137635953 EC50 > 10000 nM T42392 C5Q6ZI 137638800 Ki = 5000 nM T42392 CYI1Q0 137640284 EC50 = 390 nM T42392 C8WT0M 137640367 EC50 = 15595.53 nM T42392 C2PN1O 137640899 EC50 = 18700 nM T42392 C85CXZ 137641078 EC50 = 15595.53 nM T42392 CD53FY 137641861 EC50 = 5900 nM T42392 C4EWF7 137643689 Ki = 50000 nM T42392 C45QVR 137645605 EC50 = 950 nM T42392 CY49HW 137655786 EC50 = 10000 nM T42392 CKF3W6 137660839 Ki = 3000 nM T42392 CQG3K6 145976409 EC50 = 403300 nM T42392 C03KAU 155519563 EC50 > 1000000 nM T42392 CLWI30 145969 Ki = 108 nM T42392 D01BAG 16125102 IC50 > 100000 nM T42392 D01DMS 447196 Ki = 176 nM T42392 D03RGP 1221 Ki = 17 nM T42392 D04SMQ 440053 Ki = 898 nM T42392 D09LXQ 126569 Ki = 25.1 nM T42392 D09VYB 6420161 IC50 > 300000 nM T42392 D0J1PG 46237944 EC50 = 9332.54 nM T42392 D0K5UI 6420160 IC50 > 100000 nM T42392 D0N1CL 9799478 IC50 > 100000 nM T42392 D0T1MK 656723 Ki > 100000 nM T42392 D0T5SU 158397 Ki = 16.8 nM T86591 D00WCX 39042 EC50 = 7100 nM T86591 D05VIX 3463 EC50 = 59000 nM T86591 D07XGR 3339 IC50 = 1000 nM T86591 D0EJ6O 2763 EC50 = 900 nM T86591 D0G2MW 446284 IC50 = 1100 nM T86591 D0J5DC 2796 EC50 = 55000 nM T86591 D0N6RF 65999 EC50 > 10000 nM T86591 D0NF1U 64929 EC50 = 2646 nM T86591 D0O1TC 5280581 IC50 = 1400 nM T86591 D0UE9X 5280933 IC50 = 270 nM T86591 D02NHD 447458 Ki = 980 nM T86591 D03OSG 11236126 EC50 > 1000 nM T86591 D04BPS 9888484 EC50 = 2800 nM T86591 D04QIE 11526038 EC50 = 1 nM T86591 D0AX9S 446642 Ki = 2 nM T86591 D0H1NL 208901 EC50 = 37 nM T86591 D0I5IM 135449333 EC50 = 42 nM T86591 D0LW1Y 9864881 EC50 = 10 nM T86591 D0M0SS 170364 EC50 = 122 nM T86591 D0M3UT 206044 EC50 = 40 nM T86591 D0VU5M 9890879 EC50 = 5 nM T86591 D0H5FI 9958543 IC50 > 15000 nM T86591 D05HDX 9803963 EC50 = 229 nM T86591 D08LZI 9947731 EC50 = 10 nM T86591 D0B0EB 9890585 EC50 = 8.913 nM T86591 D0B8JQ 9825046 EC50 = 0.615 nM T86591 D0B9EN 10274777 EC50 = 50 nM T86591 C9RN3W 7127 EC50 = 46500 nM T86591 CSB8Q0 8215 IC50 = 30000 nM T86591 CVT2C4 10467 IC50 = 30000 nM T86591 C1GZ6P 128814 IC50 > 10000 nM T86591 C8R2WO 237084 EC50 = 25000 nM T86591 CUC68S 339720 EC50 > 10000 nM T86591 C20GQD 446758 EC50 = 360 nM T86591 C12SCN 637584 EC50 > 60000 nM T86591 CZN6S9 743974 IC50 > 25118.86 nM T86591 CER54F 1232372 EC50 = 0.16 nM T86591 C9KP6J 1285388 IC50 = 43000 nM T86591 CS7KF4 3110120 EC50 = 1.1 nM T86591 COH6I9 4287647 EC50 = 9500 nM T86591 CT29VZ 4388708 EC50 = 11400 nM T86591 CG7O6D 4433544 IC50 = 1500 nM T86591 C32LKN 4518233 IC50 = 1000 nM T86591 CH34WN 5281116 IC50 = 30000 nM T86591 C6K2GJ 5281805 EC50 = 8900 nM T86591 C75ORQ 5310669 EC50 = 23100 nM T86591 CZ0D2P 5715241 EC50 = 23100 nM T86591 CZJ84H 6102812 EC50 = 8 nM T86591 C16ZSG 6439929 IC50 = 20000 nM T86591 C1VU9T 6440462 EC50 = 12000 nM T86591 CLO7Y1 6540257 IC50 = 74 nM T86591 CJDX25 7009663 EC50 = 83400 nM T86591 CGXH64 9547900 EC50 = 14 nM T86591 C50PDQ 9549255 EC50 > 10000 nM T86591 C3CXT4 9802192 EC50 = 78 nM T86591 C5PGB8 9803821 EC50 = 20 nM T86591 C7TMX8 9805639 EC50 = 986 nM T86591 CCMF21 9806390 EC50 > 90000 nM T86591 C9R7OA 9822722 Ki = 72 nM T86591 C15LTP 9822765 EC50 = 20 nM T86591 CQK19U 9822766 EC50 = 40 nM T86591 CVYQ15 9822877 EC50 = 230 nM T86591 C47ZRD 9823501 EC50 = 3000 nM T86591 CXB52G 9825302 EC50 = 20 nM T86591 CSY86D 9825523 EC50 = 20 nM T86591 CJF2M6 9826186 EC50 = 6 nM T86591 C1RB9C 9842601 EC50 = 3000 nM T86591 CD04KR 9844059 EC50 = 11700 nM T86591 CG68EO 9844373 EC50 = 2900 nM T86591 CSZ36U 9844554 EC50 = 30 nM T86591 C0Z2DQ 9845736 EC50 = 90 nM T86591 C9RM5A 9845832 EC50 = 1700 nM T86591 CP5MW0 9847836 EC50 = 790 nM T86591 C6ABL9 9850395 EC50 = 8 nM T86591 C7S3YF 9866595 Ki = 560 nM T86591 CD4RY0 9867298 EC50 = 9500 nM T86591 C70MKO 9868387 EC50 = 9000 nM T86591 C7VLA1 9869022 EC50 = 1200 nM T86591 CWJU60 9870703 EC50 = 8600 nM T86591 CJ3AD7 9888213 EC50 = 110 nM T86591 C5GA7U 9888528 EC50 = 740 nM T86591 C7CB6G 9893080 EC50 = 4 nM T86591 C6O1SV 9895808 EC50 = 620 nM T86591 CY9O3C 9902264 EC50 = 60 nM T86591 C0NI1K 9908951 EC50 = 12500 nM T86591 C62YXO 9910188 EC50 > 10000 nM T86591 C57LHY 9910951 IC50 = 28 nM T86591 C7W8VE 9924989 EC50 = 620 nM T86591 CKYG10 9930277 EC50 = 300 nM T86591 C57EPL 9931070 EC50 = 670 nM T86591 C75NOF 9932563 EC50 = 3200 nM T86591 C9PCJ5 9932790 EC50 = 2500 nM T86591 CGV83S 9933541 EC50 = 6 nM T86591 CF7P8W 9934050 EC50 = 3000 nM T86591 C4VKF5 9934858 EC50 = 1900 nM T86591 C8OQX3 9935996 EC50 = 618 nM T86591 CPUF90 9952559 EC50 = 240 nM T86591 CPMH16 9953945 EC50 = 3200 nM T86591 C2VHT3 9955922 EC50 = 138 nM T86591 CRE2W1 9956726 EC50 = 4 nM T86591 C02YNS 9956737 EC50 = 240 nM T86591 C5R9BK 9959189 EC50 = 30 nM T86591 CQP9I8 9960726 EC50 = 300 nM T86591 CVM8I3 9973559 EC50 = 14000 nM T86591 CJA73Y 9980571 EC50 = 6780 nM T86591 CV74OZ 9980586 EC50 = 130 nM T86591 CFKD10 9981617 EC50 = 2 nM T86591 CF0SR7 9982519 EC50 = 3 nM T86591 C27AED 9982759 EC50 = 1350 nM T86591 CJOV70 9983904 EC50 = 150 nM T86591 C0GBI5 9985365 EC50 = 14 nM T86591 CH7W9P 10003213 EC50 = 1250 nM T86591 CKJ83Z 10004270 EC50 = 5 nM T86591 C8JV7T 10004390 Ki = 7 nM T86591 CUE80O 10004438 EC50 > 10000 nM T86591 C6VP7J 10005230 EC50 = 3 nM T86591 CK24FM 10005763 EC50 = 526 nM T86591 C6C9SG 10005877 EC50 = 200 nM T86591 C0OED7 10023279 EC50 = 350 nM T86591 C45ZDO 10026148 EC50 = 421 nM T86591 C64EJL 10027350 IC50 = 209 nM T86591 C0RVG2 10027920 EC50 = 3090 nM T86591 CLK7R6 10028864 EC50 = 170 nM T86591 C7H4RX 10050194 EC50 = 1390 nM T86591 CQH15A 10053715 EC50 > 10000 nM T86591 C48JGT 10070650 EC50 = 830 nM T86591 CNS96V 10072967 EC50 = 730 nM T86591 CCG14W 10073789 EC50 = 1130 nM T86591 CJRY94 10074505 EC50 = 560 nM T86591 CC72JH 10074964 EC50 = 175 nM T86591 C79TZB 10075037 EC50 = 1690 nM T86591 CO2IN7 10075041 EC50 = 61 nM T86591 C9PH1M 10075336 EC50 = 197 nM T86591 CR01QE 10076802 EC50 = 60 nM T86591 CL53DC 10091852 EC50 = 7470 nM T86591 CM5EU7 10093355 EC50 = 490 nM T86591 C3ZT0K 10096907 IC50 = 352 nM T86591 CQ2EH0 10096908 EC50 = 20 nM T86591 CRJU50 10098103 EC50 = 4 nM T86591 C8BWY7 10109101 EC50 = 300 nM T86591 C4FZX9 10110745 EC50 = 750 nM T86591 CI5E6O 10112797 EC50 = 354 nM T86591 CZU39A 10113515 EC50 = 2622 nM T86591 C94TCV 10113516 EC50 = 8500 nM T86591 CW5KR2 10113686 EC50 = 80 nM T86591 CQG9E4 10113721 EC50 = 8.8 nM T86591 CWH2U3 10113980 EC50 = 4 nM T86591 CL7TY9 10114135 EC50 = 127 nM T86591 C1BA8V 10114442 EC50 = 9 nM T86591 C6FIV9 10115344 IC50 = 1686 nM T86591 C1EOY3 10116365 IC50 > 50000 nM T86591 C15GVJ 10116451 EC50 = 6300 nM T86591 CY73BR 10117908 EC50 > 10000 nM T86591 CTGB91 10118056 EC50 = 120 nM T86591 CRCG14 10118927 Ki = 1100 nM T86591 CFZ80V 10119392 EC50 = 69 nM T86591 C98ENV 10119393 EC50 = 7 nM T86591 CU89OW 10119824 EC50 = 900 nM T86591 C3RDM7 10136188 EC50 = 130 nM T86591 CWGV68 10136347 EC50 = 111 nM T86591 C74VJE 10136660 EC50 = 1880 nM T86591 C8O0AV 10137115 EC50 = 336 nM T86591 C2N6UZ 10137230 IC50 > 3300 nM T86591 CEN20X 10137337 EC50 = 30 nM T86591 CDX37J 10137693 EC50 = 6 nM T86591 CVI26N 10138146 EC50 = 10 nM T86591 CMRP39 10139247 EC50 = 12 nM T86591 CB3SH2 10139551 EC50 = 240 nM T86591 C6RPI1 10139836 EC50 = 50 nM T86591 C6N1TJ 10140233 EC50 = 5 nM T86591 CBE62A 10140247 EC50 = 171 nM T86591 CR4E1D 10141305 EC50 = 240 nM T86591 CB53WS 10141607 IC50 = 48 nM T86591 C0OD9X 10141609 EC50 = 2800 nM T86591 CQM84R 10142329 EC50 = 23 nM T86591 C78OLG 10143678 EC50 = 845 nM T86591 CW04MX 10144243 EC50 = 78 nM T86591 CD73IB 10157036 EC50 = 3 nM T86591 CIXB29 10157662 EC50 = 202 nM T86591 CKH28L 10157940 EC50 = 9975 nM T86591 C7XT5K 10159635 EC50 = 40 nM T86591 C4XM1D 10160128 EC50 = 199 nM T86591 C05LIH 10161760 EC50 = 82 nM T86591 C4T7GE 10161854 Ki = 14 nM T86591 C95FYK 10161996 EC50 = 75 nM T86591 C9C3JQ 10162008 EC50 = 2 nM T86591 CZ24HT 10162063 EC50 = 4 nM T86591 C7DU6F 10162210 EC50 = 80 nM T86591 CDM26O 10162519 EC50 = 40 nM T86591 CMF69H 10162615 IC50 = 5800 nM T86591 C6JB5Q 10162929 EC50 = 58 nM T86591 C6AE1Y 10163556 EC50 = 110 nM T86591 CFE2M9 10163810 EC50 = 4000 nM T86591 CZ6EW0 10164032 EC50 > 30000 nM T86591 CM21IJ 10164033 IC50 = 529 nM T86591 C9FR3O 10174350 IC50 = 4.699 nM T86591 C2RL8N 10177074 EC50 = 100 nM T86591 CH34CD 10177349 EC50 = 30 nM T86591 C93CIF 10177377 Ki = 38 nM T86591 CO1Y3R 10178534 EC50 = 10 nM T86591 C5JHK0 10181314 EC50 = 38 nM T86591 C52QCT 10182727 EC50 = 104 nM T86591 CDT75W 10182946 EC50 = 2 nM T86591 CUQ89L 10183490 EC50 = 31 nM T86591 C49HSN 10183977 EC50 = 22 nM T86591 C7V1ML 10186118 EC50 = 45 nM T86591 C89CVS 10186123 EC50 > 10000 nM T86591 CFCY37 10186986 EC50 = 6456.54 nM T86591 CDF82U 10199589 EC50 = 890 nM T86591 CPW69C 10199828 EC50 = 1300 nM T86591 CPM13H 10201545 EC50 = 10 nM T86591 CVD5N1 10202000 EC50 = 182 nM T86591 C7NPZ3 10202354 Ki = 15 nM T86591 CJ0R3W 10202547 EC50 = 3280 nM T86591 C1J2VR 10204076 EC50 = 65 nM T86591 CC3G0I 10204762 EC50 = 36 nM T86591 CYA5S6 10204908 EC50 = 2700 nM T86591 CY1ZK2 10205220 EC50 = 70 nM T86591 C0F5CK 10205615 EC50 = 58 nM T86591 CAQ5U8 10205828 IC50 = 3300 nM T86591 CMSG62 10207241 EC50 = 20 nM T86591 C6MYJ4 10207242 EC50 = 6100 nM T86591 CM4HS7 10207244 EC50 = 700 nM T86591 C27EYG 10207287 EC50 > 10000 nM T86591 CO52SH 10208214 EC50 = 4600 nM T86591 C03WGI 10208599 Ki = 19 nM T86591 CJF3K8 10210559 EC50 = 49 nM T86591 C1NIA4 10217191 IC50 = 482 nM T86591 CPAH95 10222749 EC50 = 10001 nM T86591 CL1K2N 10223023 IC50 = 567.54 nM T86591 C9VEU1 10223369 EC50 = 1573 nM T86591 C9SIT0 10223583 IC50 = 877 nM T86591 CI57ZX 10223837 EC50 = 271 nM T86591 CS25KJ 10224123 EC50 = 37 nM T86591 CY28GC 10224783 EC50 = 24 nM T86591 C4R7LT 10224945 EC50 = 254 nM T86591 CQ56VG 10225637 EC50 = 7 nM T86591 CU1T0A 10225684 EC50 = 119 nM T86591 CJH81C 10225731 EC50 = 220 nM T86591 C2RY6K 10225793 EC50 = 354 nM T86591 CYR3B5 10226233 EC50 = 2870 nM T86591 CG4P7X 10226511 EC50 = 120 nM T86591 CUS8V5 10227653 EC50 > 15000 nM T86591 CS7Q9U 10229225 EC50 = 10 nM T86591 C1UF8K 10232157 EC50 = 260 nM T86591 COVB68 10252612 IC50 = 73 nM T86591 CC8GU0 10254028 EC50 = 254 nM T86591 CARH74 10254209 EC50 = 170 nM T86591 C2HIT7 10254845 IC50 = 40 nM T86591 C3OE5Z 10257392 EC50 = 40 nM T86591 C9KZJ3 10270710 EC50 = 20000 nM T86591 CVH34N 10274499 EC50 = 109 nM T86591 C4PM2S 10274627 EC50 = 2000 nM T86591 CR6L1U 10274642 EC50 = 61 nM T86591 CH59WA 10274664 EC50 = 559 nM T86591 CJCU12 10274955 EC50 = 92 nM T86591 CZ64AI 10275334 EC50 = 10 nM T86591 C72YHL 10275376 EC50 = 5600 nM T86591 C73ZHW 10276052 Ki = 10 nM T86591 CI1BV7 10276470 IC50 > 15000 nM T86591 C7YMO1 10276539 Ki = 4 nM T86591 CIOK04 10277666 EC50 = 30 nM T86591 C02EHS 10279905 IC50 = 3900 nM T86591 CW34DF 10280116 EC50 = 4 nM T86591 CSJ28C 10280496 IC50 = 2770 nM T86591 CS1U0K 10281422 IC50 > 15000 nM T86591 CW9HU6 10288123 EC50 = 1210 nM T86591 CC5K1M 10292707 IC50 = 230 nM T86591 CEI98Y 10294076 EC50 = 6000 nM T86591 CCN93S 10294697 EC50 = 130 nM T86591 CQR18V 10295993 EC50 = 5640 nM T86591 CY28SU 10296059 EC50 = 12000 nM T86591 CP2MO0 10296330 EC50 = 5700 nM T86591 CK7F1O 10297427 EC50 = 28 nM T86591 CO1P5R 10297760 EC50 = 2152 nM T86591 CL40QG 10297943 EC50 = 30 nM T86591 CXA6K2 10298514 EC50 = 300 nM T86591 CLE54O 10298859 EC50 = 53 nM T86591 CL5WB3 10299983 EC50 = 4 nM T86591 CS9V4N 10300072 EC50 = 5200 nM T86591 C89QXN 10300073 IC50 = 2000 nM T86591 C7UNX1 10300279 EC50 = 4 nM T86591 CLQD46 10301814 EC50 = 210 nM T86591 CFS25Z 10320822 EC50 = 50 nM T86591 CQH6P7 10323352 EC50 = 328 nM T86591 CDU6H7 10323599 EC50 = 180 nM T86591 C7S4LC 10324316 EC50 = 9 nM T86591 CGD4N7 10341169 EC50 = 840 nM T86591 C01MTP 10341401 EC50 = 70 nM T86591 CG58VR 10341444 EC50 = 1500 nM T86591 C46JQA 10341445 EC50 = 60 nM T86591 C6HM5O 10342769 EC50 = 70 nM T86591 C8AT6R 10342801 EC50 = 9 nM T86591 C3NJ4S 10343538 EC50 = 410 nM T86591 CB6R4D 10344769 EC50 = 30 nM T86591 CPO38A 10345547 EC50 = 20 nM T86591 C92PZC 10346786 EC50 = 1 nM T86591 CPT82D 10347115 EC50 = 140 nM T86591 CR5P7Z 10347250 EC50 = 8 nM T86591 C0OP5K 10347566 EC50 = 30 nM T86591 C23JXU 10367018 EC50 = 2 nM T86591 C84KIW 10367602 IC50 = 237 nM T86591 C0SKH9 10368050 EC50 = 8 nM T86591 CMW4U5 10368444 EC50 = 44 nM T86591 CDA5F7 10369999 EC50 = 40 nM T86591 CB8KU1 10370056 EC50 = 10 nM T86591 CC1IK3 10370262 EC50 > 10000 nM T86591 C0SLF7 10371709 EC50 = 710 nM T86591 CN92GI 10387634 EC50 = 13 nM T86591 C8LG4Z 10390333 EC50 = 6 nM T86591 CLI13C 10390756 EC50 = 641 nM T86591 CJQV19 10391684 EC50 = 70 nM T86591 C7PO5N 10392711 Ki < 3019.95 nM T86591 CTMS40 10409008 EC50 = 10000 nM T86591 CQY70C 10409988 EC50 = 1000 nM T86591 C9GLW7 10410878 EC50 = 40 nM T86591 CJB86G 10411897 IC50 = 175 nM T86591 C29PFI 10412116 EC50 = 90 nM T86591 C5AWB0 10414708 EC50 = 74 nM T86591 CBN4H0 10415698 EC50 = 5 nM T86591 C72JHZ 10432356 IC50 = 121 nM T86591 CEO2U1 10432525 EC50 = 43 nM T86591 CTQ0R7 10433053 EC50 = 1000 nM T86591 CKGE28 10434749 EC50 = 10000 nM T86591 C63QBA 10455509 EC50 = 190 nM T86591 CWQ2K1 10455511 EC50 = 20 nM T86591 CT7PM6 10455681 EC50 = 1140 nM T86591 C1S7GU 10455871 EC50 = 5800 nM T86591 C4DXE1 10457843 EC50 = 53 nM T86591 C1H5RP 10458842 EC50 = 5 nM T86591 C05UYW 10460941 Ki < 3019.95 nM T86591 C9Q5HV 10480558 EC50 = 170 nM T86591 CJ6S2A 10480923 EC50 = 105 nM T86591 CP04MX 10481007 EC50 = 150 nM T86591 CGXY36 10482372 EC50 = 10 nM T86591 CL69EZ 10507132 Ki = 125.89 nM T86591 CR1O9Z 10531248 Ki = 107.15 nM T86591 C9GJD6 10554575 Ki = 173.78 nM T86591 CJ2O0B 10554759 Ki < 3019.95 nM T86591 C04RCN 10554988 Ki = 467.74 nM T86591 CU8QT4 10578478 Ki < 3019.95 nM T86591 CY4F5V 10578925 Ki = 177.83 nM T86591 C1B8PZ 10602637 Ki = 138.04 nM T86591 CZG3C2 10626761 Ki < 3019.95 nM T86591 C6GV9A 10674474 Ki = 56.23 nM T86591 CMTU60 10674509 Ki = 45.71 nM T86591 CBL6H3 10674589 Ki < 3019.95 nM T86591 C4PIH1 10698305 Ki = 1905.46 nM T86591 CPZG21 10721272 Ki = 407.38 nM T86591 C26MKN 10723133 Ki < 3019.95 nM T86591 C8KNR9 10743135 EC50 = 1400 nM T86591 C07ANU 10746810 Ki = 2511.89 nM T86591 CGI0V4 10792302 Ki < 3019.95 nM T86591 CYE68O 10792674 Ki < 3019.95 nM T86591 CGF14Z 10793522 Ki < 3019.95 nM T86591 CP9J3U 10840584 Ki = 1862.09 nM T86591 CZG96J 10896097 EC50 > 50000 nM T86591 CFW9J2 10896153 EC50 = 2398.83 nM T86591 C5J4PX 10896495 EC50 > 50000 nM T86591 CYI87W 10914801 EC50 = 2300 nM T86591 C9PIM1 10916251 EC50 = 4900 nM T86591 CJ50OD 10939255 EC50 = 1500 nM T86591 C6UIW4 10983398 EC50 = 61.9 nM T86591 C80VSA 10992201 EC50 = 625 nM T86591 C5BN4L 11024616 EC50 = 2751 nM T86591 CJBM20 11042473 EC50 = 15700 nM T86591 CF38JZ 11048469 EC50 = 1600 nM T86591 CRK95E 11049998 EC50 = 218.78 nM T86591 CSJ7R0 11058026 EC50 = 500 nM T86591 CG23SM 11071056 EC50 = 42900 nM T86591 CV7UL0 11090513 EC50 = 860 nM T86591 CZD8U3 11101345 EC50 = 680 nM T86591 CR26YH 11111473 EC50 = 1200 nM T86591 CX6IM8 11122999 EC50 = 2800 nM T86591 C8E4YR 11133305 EC50 = 320 nM T86591 C5KB7N 11153268 EC50 = 250 nM T86591 C61TQH 11154732 EC50 > 1000 nM T86591 CQ13LJ 11155087 EC50 = 2850 nM T86591 CG2V4U 11155122 EC50 = 70 nM T86591 CIV54T 11155356 EC50 > 1000 nM T86591 C3LG4F 11155783 EC50 = 8 nM T86591 CP9NX6 11156185 EC50 = 2200 nM T86591 CN47MW 11165712 EC50 = 48 nM T86591 CLA09R 11165781 IC50 = 3900 nM T86591 CN7QF3 11166818 EC50 = 20 nM T86591 CIW98T 11167613 EC50 = 20 nM T86591 CF0H2Q 11167738 EC50 = 32 nM T86591 C3OWD7 11169884 EC50 = 6690 nM T86591 CSO27I 11177525 IC50 = 800 nM T86591 C4W7XI 11178006 EC50 = 2870 nM T86591 C6IZ7D 11178075 IC50 = 89 nM T86591 C1M9TC 11178156 EC50 = 290 nM T86591 CW2FH7 11178750 EC50 = 1 nM T86591 CM3BO2 11178916 EC50 = 75 nM T86591 C6BQ7O 11179502 EC50 = 90 nM T86591 CY3LO2 11184855 EC50 = 2500 nM T86591 C01XFA 11186225 EC50 = 3900 nM T86591 C3EGQ4 11186282 EC50 = 10 nM T86591 CXA72P 11188236 EC50 = 160 nM T86591 CK84AR 11188766 IC50 = 3820 nM T86591 C50QOG 11189474 IC50 = 393 nM T86591 C8EIV0 11189652 IC50 = 1410 nM T86591 C2D9FS 11190667 EC50 = 4 nM T86591 CA7K4Q 11190685 EC50 > 1000 nM T86591 C7B0QN 11190733 EC50 = 100 nM T86591 CQ42YC 11199906 EC50 = 83 nM T86591 C89UCH 11202658 EC50 = 30 nM T86591 C2JK4F 11203145 EC50 = 130 nM T86591 CYHZ54 11208735 EC50 = 24550 nM T86591 C7ZPE1 11211156 EC50 > 1000 nM T86591 C71NVH 11211999 EC50 = 1890 nM T86591 CO73VY 11212480 EC50 = 110 nM T86591 CU2F0D 11213609 EC50 = 3.5 nM T86591 C7P2LF 11214000 EC50 > 10000 nM T86591 C3G7FR 11214539 EC50 = 28 nM T86591 CM6I2B 11218775 EC50 = 8317.64 nM T86591 C7S9CH 11223211 EC50 = 76 nM T86591 C92VLZ 11223613 IC50 = 23 nM T86591 C8JZ6Q 11225048 EC50 = 2 nM T86591 C8ATL5 11225797 EC50 = 474 nM T86591 CJ78RY 11225851 EC50 = 97 nM T86591 CE4I3N 11225910 EC50 > 1000 nM T86591 CD2NX7 11227195 EC50 = 570 nM T86591 CQJ5E6 11234410 EC50 = 3140 nM T86591 C2JNM9 11234452 EC50 = 670 nM T86591 CBSO15 11234869 EC50 = 144 nM T86591 C7ROX3 11235560 EC50 = 2890 nM T86591 CQ3C1F 11235892 EC50 = 186 nM T86591 CBU98W 11236923 EC50 = 8 nM T86591 CF31OJ 11237218 EC50 = 85 nM T86591 CGAI13 11237761 EC50 > 3000 nM T86591 C3B5FX 11243082 EC50 = 13489.63 nM T86591 CG8IQ1 11246863 EC50 > 1000 nM T86591 CL29MP 11247579 EC50 = 19 nM T86591 CP1X0G 11247654 EC50 = 2980 nM T86591 C7C9MZ 11247664 EC50 = 468 nM T86591 CBS49N 11247908 EC50 = 383 nM T86591 CY10BP 11247998 IC50 = 150 nM T86591 C5VB4A 11248512 EC50 = 2 nM T86591 C79VCR 11249385 IC50 = 3000 nM T86591 C7LK0I 11258987 EC50 = 5211 nM T86591 CJ6ON0 11259787 EC50 = 94 nM T86591 CH9X1P 11260214 EC50 = 170 nM T86591 CRC0K9 11268768 EC50 = 20000 nM T86591 C9J3DR 11271060 EC50 = 549 nM T86591 C7ZC0P 11271211 EC50 = 45 nM T86591 CYD12Z 11271514 EC50 = 50 nM T86591 CWH02S 11280270 EC50 > 1000 nM T86591 CK87RJ 11281114 EC50 = 260 nM T86591 CH69MT 11281802 EC50 = 115 nM T86591 C2O3WX 11283113 EC50 = 730 nM T86591 CP0H1J 11293283 EC50 > 1000 nM T86591 CDK79P 11293459 EC50 > 3000 nM T86591 C6T9OR 11294565 EC50 = 270 nM T86591 C5S6YO 11294660 EC50 > 10000 nM T86591 CFTW52 11295349 EC50 = 544 nM T86591 CMC6I8 11305717 EC50 = 1529 nM T86591 CC81HS 11306364 IC50 = 1047.13 nM T86591 CDKC74 11306495 EC50 > 3000 nM T86591 C2KZ3M 11306745 EC50 = 42 nM T86591 CB12CE 11316788 EC50 = 2813 nM T86591 C7Z1NC 11317347 EC50 = 476 nM T86591 CUW3Q0 11317867 EC50 = 561 nM T86591 C0D7HU 11317892 IC50 > 15000 nM T86591 CFQV09 11323235 EC50 = 28700 nM T86591 CUSY83 11327370 IC50 = 550 nM T86591 CHO5P0 11327951 IC50 = 261 nM T86591 C1OEB0 11328910 EC50 = 2888 nM T86591 C9SB2M 11329011 EC50 = 186 nM T86591 CSF2L4 11329304 EC50 = 45 nM T86591 CUL9I0 11335874 EC50 = 500 nM T86591 C6O3ZU 11339029 IC50 = 34 nM T86591 CMCD29 11339649 EC50 > 3000 nM T86591 C6WI0Z 11339975 IC50 = 26.98 nM T86591 CP5F8D 11339979 IC50 = 72 nM T86591 C9B0LH 11340275 EC50 > 1000 nM T86591 CG91XM 11340322 EC50 = 425 nM T86591 C0ABC9 11340513 EC50 = 686 nM T86591 CLFX14 11340991 EC50 = 2558 nM T86591 C0LU6S 11349723 EC50 > 1000 nM T86591 CATM03 11350008 IC50 = 6120 nM T86591 CQ7OF6 11351221 EC50 > 1000 nM T86591 CDL72P 11351238 EC50 = 46 nM T86591 CEZG39 11351266 EC50 > 1000 nM T86591 C72GEN 11351550 EC50 = 64 nM T86591 CL7D8V 11351980 EC50 = 34 nM T86591 C9PAJ6 11352187 EC50 = 656 nM T86591 CQN0X9 11352573 EC50 = 921 nM T86591 CET87Y 11352791 EC50 > 25000 nM T86591 C8QTH7 11356973 EC50 = 3900 nM T86591 C8SYL1 11362482 EC50 = 1200 nM T86591 C8VT0Y 11362757 EC50 = 56 nM T86591 CZ30DH 11363106 EC50 = 23 nM T86591 CM7TX9 11363175 EC50 = 57 nM T86591 CXHU81 11374318 EC50 = 160 nM T86591 C81BYX 11374677 EC50 = 18 nM T86591 CKE9R8 11374679 EC50 = 10 nM T86591 CDQ2M5 11374680 EC50 = 50 nM T86591 CJI2C6 11376123 EC50 = 200 nM T86591 CZ5UX9 11381586 EC50 = 4000 nM T86591 C93MQC 11383635 IC50 > 50000 nM T86591 C5F8EY 11383668 EC50 = 1237 nM T86591 C5TZY0 11385663 EC50 = 37 nM T86591 C3Z1LN 11386159 EC50 = 33 nM T86591 C8WVM5 11386220 EC50 = 2 nM T86591 C5OB8J 11386857 EC50 = 206 nM T86591 C8X5PW 11393977 EC50 = 10 nM T86591 C6SYD8 11396352 EC50 > 1000 nM T86591 CTU8G6 11397018 EC50 = 9 nM T86591 C0TX7O 11397203 EC50 = 94 nM T86591 CXIN63 11397705 EC50 = 1 nM T86591 COK68W 11399560 EC50 = 80 nM T86591 CGY28A 11405204 EC50 > 1000 nM T86591 CZB52S 11408244 IC50 = 1016 nM T86591 C34QBC 11408475 EC50 = 389.05 nM T86591 CX7W4S 11408502 EC50 = 41 nM T86591 CPB8F6 11409173 EC50 = 2630 nM T86591 CVG1X9 11414728 EC50 = 10900 nM T86591 C45UNR 11416269 IC50 > 10000 nM T86591 CKGU54 11418373 IC50 > 15000 nM T86591 CCAJ14 11418941 EC50 > 1000 nM T86591 C6Q8FR 11419459 EC50 = 10 nM T86591 CXJ72D 11419635 IC50 = 230 nM T86591 C2USN6 11419919 IC50 = 130 nM T86591 CI6ZE4 11419960 IC50 = 790 nM T86591 CMT65A 11421645 EC50 > 1000 nM T86591 CCD7X1 11421714 EC50 = 2393 nM T86591 CZ3VT9 11430761 EC50 = 15 nM T86591 C60KVM 11431103 EC50 = 877 nM T86591 C5SKD2 11431192 EC50 = 67 nM T86591 CPGX09 11431289 EC50 = 79 nM T86591 C1OZ5D 11431625 EC50 = 37 nM T86591 CFU62G 11432162 EC50 = 66 nM T86591 C8XQL7 11438721 EC50 = 900 nM T86591 C6FP3T 11441763 EC50 > 1000 nM T86591 CT4NR0 11442228 EC50 > 1000 nM T86591 C2ZVF9 11442294 EC50 = 4 nM T86591 CV5M3A 11442379 EC50 = 504 nM T86591 CKF91A 11448976 IC50 > 50000 nM T86591 CO5M3W 11449787 IC50 = 3000 nM T86591 CE59YF 11453821 EC50 = 11.5 nM T86591 C6Q7UX 11454132 EC50 = 2700 nM T86591 C04YQX 11454155 EC50 = 4 nM T86591 CR5LM7 11463604 EC50 = 882 nM T86591 CJ7RT2 11463615 IC50 = 130 nM T86591 C7XLZ9 11463785 EC50 = 105 nM T86591 C2Q6YV 11463996 IC50 > 50000 nM T86591 CF63PO 11464352 EC50 = 78 nM T86591 C4ZE1C 11465146 EC50 = 94 nM T86591 CQT9S6 11466042 EC50 = 310 nM T86591 CW7U6D 11471872 EC50 = 1400 nM T86591 C6G7FO 11475460 EC50 > 1000 nM T86591 CN64KX 11475461 EC50 > 1000 nM T86591 C0V4HX 11476137 EC50 = 90 nM T86591 C7ZO8B 11476297 EC50 > 1000 nM T86591 CLZ5I1 11476382 EC50 > 3000 nM T86591 CI8FO6 11476916 EC50 = 100 nM T86591 CSX3Z0 11477433 EC50 > 25000 nM T86591 C83GWX 11477735 EC50 = 736 nM T86591 CQ6L9S 11486733 EC50 > 1000 nM T86591 C4S6JR 11488006 EC50 > 1000 nM T86591 CZ84QA 11488726 EC50 = 2654 nM T86591 C6HO8J 11490050 EC50 > 1000 nM T86591 CQ9P3C 11497430 EC50 = 114 nM T86591 CL2V9K 11497604 EC50 > 10000 nM T86591 CF1AI0 11503439 EC50 = 5 nM T86591 CU27FT 11503588 EC50 = 311 nM T86591 CF36HJ 11508312 EC50 > 10000 nM T86591 C0JEO8 11511317 IC50 = 1079 nM T86591 CL4N9S 11512673 EC50 > 100000 nM T86591 C68RSH 11525752 IC50 = 450 nM T86591 CCJ50E 11526339 EC50 = 11130 nM T86591 CH14EK 11526493 EC50 = 19 nM T86591 CU5A2J 11532616 EC50 = 1200 nM T86591 CT9Z0X 11539510 EC50 = 250 nM T86591 C52AIP 11546956 IC50 = 10575 nM T86591 C5H7FP 11563028 IC50 > 50000 nM T86591 C9SJL1 11570226 EC50 > 100000 nM T86591 CF2V1D 11583815 IC50 = 4486 nM T86591 C3GI8R 11585006 EC50 > 10000 nM T86591 CD6W0Y 11588094 EC50 > 10000 nM T86591 C1HG4A 11591164 IC50 > 50000 nM T86591 CC15AQ 11592357 IC50 > 50000 nM T86591 CDR1Z3 11599646 EC50 = 12 nM T86591 C2ZP9O 11612623 EC50 = 1819 nM T86591 CE87MQ 11619439 EC50 = 5 nM T86591 C5LVA3 11620018 EC50 = 2 nM T86591 C4M5SU 11620299 EC50 > 1000 nM T86591 CWOD63 11620575 IC50 > 50000 nM T86591 CQN62W 11626766 IC50 = 780 nM T86591 CR30AV 11627288 EC50 = 50 nM T86591 C4ZR8D 11627859 EC50 = 1310 nM T86591 C1GD3M 11628577 EC50 = 1350 nM T86591 CA1U4D 11630055 EC50 = 1800 nM T86591 C1FI8K 11635845 EC50 = 1450 nM T86591 CM6R1L 11640895 IC50 = 116 nM T86591 C6QZ4F 11649387 EC50 = 8980 nM T86591 C16CWN 11649783 EC50 = 3330 nM T86591 CY2DE9 11656305 EC50 = 2200 nM T86591 C9H2TQ 11660029 EC50 > 10000 nM T86591 CD0NU7 11663038 EC50 = 500 nM T86591 CL7C1Z 11663931 EC50 > 10000 nM T86591 CQ2M8V 11669781 IC50 = 399.94 nM T86591 C1OH3U 11674387 EC50 = 1632 nM T86591 C27FGM 11677450 EC50 = 18 nM T86591 CHA36Y 11678044 EC50 = 2475 nM T86591 C6H8PJ 11678481 EC50 = 790 nM T86591 C91EWR 11678534 IC50 > 50000 nM T86591 C2CHW3 11682417 EC50 = 1142 nM T86591 C8MU1C 11683336 EC50 = 10 nM T86591 CS3PO8 11698476 EC50 = 760 nM T86591 CD43TA 11698802 IC50 > 50000 nM T86591 C3FIK4 11704026 EC50 = 160 nM T86591 C7P8FY 11704978 IC50 = 8300 nM T86591 CGK13J 11705301 IC50 = 4400 nM T86591 CR46YH 11705832 IC50 = 414 nM T86591 C2WQ1O 11711595 EC50 = 10 nM T86591 C5AX8M 11712774 EC50 = 169 nM T86591 C2UY7P 11712873 EC50 = 1037 nM T86591 CJU3Z2 11716196 EC50 = 35900 nM T86591 CLF57E 11729251 EC50 = 1800 nM T86591 C5UIL7 11729738 EC50 = 400 nM T86591 C6C9HF 11741962 IC50 = 125 nM T86591 C5FYH0 11742116 EC50 = 140 nM T86591 CNQ6O1 11750720 EC50 > 1000 nM T86591 C51EZG 11750812 IC50 = 260 nM T86591 CR7Y2E 11751021 EC50 = 2680 nM T86591 C7V0DE 11751301 EC50 = 4.9 nM T86591 C0Q4XH 11753952 EC50 = 5 nM T86591 C35DKP 11754345 EC50 = 83 nM T86591 CLE5P8 11754583 EC50 = 130 nM T86591 C7O6FH 11755396 EC50 = 520 nM T86591 C18XBA 11755655 EC50 = 37 nM T86591 CL4EK8 11755968 EC50 = 87 nM T86591 C58DMZ 11757696 EC50 = 8 nM T86591 C13LEO 11760451 EC50 = 9400 nM T86591 CKWA01 11772573 IC50 = 1600 nM T86591 CPV6E2 11774184 EC50 = 226 nM T86591 C9D4OH 11774537 EC50 = 91 nM T86591 C7WQ9E 11774595 EC50 = 39 nM T86591 CBV25C 11774828 EC50 = 2880 nM T86591 C95FTM 11774965 EC50 = 2800 nM T86591 CE27GQ 11775099 EC50 = 833 nM T86591 C3EXH7 11775225 EC50 > 10000 nM T86591 CA0LW8 11784454 EC50 = 140 nM T86591 CX5YP8 11784860 EC50 = 10 nM T86591 CW8R9F 11785036 EC50 = 34 nM T86591 CHUA47 11801489 Ki < 3019.95 nM T86591 CU01OH 11810803 EC50 = 3100 nM T86591 C5N4VH 11811337 EC50 = 2200 nM T86591 C5MJ8U 11811825 EC50 = 9600 nM T86591 CL7V4Z 11826628 EC50 = 410 nM T86591 CAO2Q1 11948655 EC50 = 96 nM T86591 CUJ2S3 11954219 IC50 = 240 nM T86591 C38KZG 11978565 EC50 = 8700 nM T86591 CEW4G1 11978566 EC50 = 7700 nM T86591 CQH67B 11978567 EC50 = 7000 nM T86591 C1AOP8 11978570 EC50 = 2300 nM T86591 CN2S4P 11982685 EC50 = 3200 nM T86591 C1CBW0 11992126 EC50 = 173 nM T86591 COPI61 11997929 EC50 > 10000 nM T86591 CV2OW5 12132847 EC50 = 181 nM T86591 C8VJ4Y 12928398 EC50 = 14300 nM T86591 CWL9C6 12967684 EC50 = 1600 nM T86591 C1LW6C 14086141 EC50 = 9300 nM T86591 CQSK24 14163455 IC50 = 1210 nM T86591 CS82RI 14427412 EC50 = 4000 nM T86591 C8X0RD 15604876 EC50 = 3500 nM T86591 C0LH2E 15942850 EC50 = 1100 nM T86591 C6J5WN 15951505 IC50 = 20 nM T86591 CF6I7X 15981441 EC50 = 790 nM T86591 CDFT16 15984029 EC50 = 1000 nM T86591 CEL3S6 16007090 EC50 = 1330 nM T86591 C9T1QR 16036021 EC50 > 10000 nM T86591 CT3VA7 16036134 EC50 > 10000 nM T86591 CWE62Y 16038358 EC50 = 7220 nM T86591 CO5B2T 16043249 EC50 > 10000 nM T86591 CY13OS 16046718 EC50 = 500 nM T86591 CTP15X 16046722 EC50 = 1000 nM T86591 CE1A9C 16058409 EC50 = 1520 nM T86591 C05RLT 16058623 EC50 = 3 nM T86591 C4ENU6 16058624 EC50 = 56 nM T86591 CD3K9X 16085980 EC50 = 1524 nM T86591 CY1Q3Z 16085981 EC50 = 642 nM T86591 C1F6CM 16085982 EC50 = 2067 nM T86591 C97HJA 16085983 EC50 = 710 nM T86591 CE3HN1 16085984 EC50 = 2929 nM T86591 C2F4AJ 16085985 EC50 = 2204 nM T86591 CE4Q7N 16085986 EC50 = 488 nM T86591 CXYF29 16085987 EC50 = 2224 nM T86591 CPQ2K9 16085988 EC50 = 2800 nM T86591 CF4J1K 16090330 EC50 = 1300 nM T86591 CU63PB 16090857 EC50 = 32 nM T86591 CA51QP 16090858 EC50 = 282 nM T86591 C8O1HI 16090859 EC50 = 1099 nM T86591 CMKI28 16090878 EC50 = 2078 nM T86591 CJC53L 16090879 EC50 = 120 nM T86591 C3E6XL 16103189 EC50 > 10000000 nM T86591 C0AOB9 16103190 EC50 > 10000000 nM T86591 CI53BG 16103191 EC50 = 11000 nM T86591 C4ENB3 16103192 EC50 = 21000 nM T86591 CJ3D4H 16109183 EC50 = 210 nM T86591 CJ38DY 16109187 EC50 = 9500 nM T86591 CS8NF6 16109190 EC50 = 70 nM T86591 C9IO5Z 16109193 EC50 = 4 nM T86591 CU0BK1 16109199 EC50 = 1320 nM T86591 C2S0TO 16109209 EC50 = 465 nM T86591 C7V9EL 16109210 EC50 > 10000 nM T86591 CP0SB8 16110418 EC50 > 10000 nM T86591 C4W5IY 16110419 EC50 = 1610 nM T86591 CHJ4Z3 16110420 EC50 > 10000 nM T86591 C2TO3Q 16110421 EC50 > 10000 nM T86591 C2KPE7 16110422 EC50 > 10000 nM T86591 CE16PQ 16110423 EC50 > 10000 nM T86591 CDVL80 16110424 EC50 = 9360 nM T86591 C3X2WM 16110425 EC50 = 3950 nM T86591 C4T0RO 16110426 EC50 > 10000 nM T86591 CT78IG 16110427 EC50 = 7500 nM T86591 CYZ74P 16110428 EC50 > 10000 nM T86591 C7IL6H 16110429 EC50 = 6850 nM T86591 CE91XP 16110436 EC50 > 10000 nM T86591 C9W4KS 16110437 EC50 = 3270 nM T86591 C2OZJ4 16110438 EC50 = 6600 nM T86591 C6FA1K 16110439 EC50 = 1690 nM T86591 CI05UK 16110440 EC50 > 10000 nM T86591 CI4Z8S 16110441 EC50 = 7280 nM T86591 C2UJ6Y 16110442 EC50 > 10000 nM T86591 CBW78Z 16110443 EC50 = 5260 nM T86591 CE19FD 16110444 EC50 = 2900 nM T86591 C7F0IX 16110482 EC50 = 111 nM T86591 C3PXV5 16110483 EC50 = 255 nM T86591 C5WZ4Y 16110484 EC50 = 268 nM T86591 CCM5G9 16110485 EC50 = 1280 nM T86591 C0N6VP 16110486 EC50 = 147 nM T86591 C5NX0T 16110487 EC50 = 437 nM T86591 C7Q2PD 16110488 EC50 = 112 nM T86591 CC24LB 16110489 EC50 = 135 nM T86591 CNU63E 16110490 EC50 = 9901477.39 nM T86591 CHD61I 16110491 EC50 = 803 nM T86591 CQ0T9X 16110492 EC50 = 6490 nM T86591 CF15DS 16110493 EC50 = 100 nM T86591 CTC3I5 16110494 EC50 = 47 nM T86591 CNS35L 16110511 EC50 = 1980 nM T86591 CXQD14 16110512 EC50 = 6800 nM T86591 CKSV19 16110513 EC50 = 5700 nM T86591 C4TO1G 16110514 EC50 > 10000 nM T86591 CKN05Q 16110515 EC50 > 10000 nM T86591 CZ5RS7 16110516 EC50 > 10000 nM T86591 CU1S0A 16110517 EC50 = 700 nM T86591 CO5D1F 16110518 EC50 > 10000 nM T86591 CB8Q6G 16110519 EC50 = 9200 nM T86591 CW4V2X 16110524 EC50 = 328 nM T86591 CT35DL 16110525 EC50 = 2530 nM T86591 C4F5EU 16110532 EC50 = 10000 nM T86591 C09TRM 16110533 EC50 = 2480 nM T86591 CZ3AN2 16110534 EC50 = 755 nM T86591 CXN40P 16110535 EC50 = 520 nM T86591 CE71MI 16220190 EC50 = 240 nM T86591 CR3C1Q 16222636 EC50 = 500 nM T86591 C49IER 16722365 EC50 = 160 nM T86591 CD7L4Z 16726113 EC50 > 1000 nM T86591 C92NRU 16727109 EC50 = 4 nM T86591 CM9YZ5 16739272 EC50 = 22 nM T86591 CN6CU3 16739344 EC50 = 1772 nM T86591 CD65RZ 16742591 EC50 = 32 nM T86591 C8LPX0 16747684 EC50 = 2 nM T86591 CCPS15 16753427 IC50 = 2200 nM T86591 C83AOY 17894227 Ki = 7.3 nM T86591 CFS4T7 17894542 EC50 = 260 nM T86591 CW4K9X 17984540 EC50 = 515 nM T86591 CW29KQ 18003431 IC50 = 69 nM T86591 CHB98X 18003446 IC50 = 61 nM T86591 C8WQ6D 18003447 IC50 = 22 nM T86591 CAOS67 18003481 IC50 = 120 nM T86591 CA32RT 18003618 EC50 = 48 nM T86591 CAO59H 18438761 EC50 = 185 nM T86591 CT1CI8 18442899 EC50 = 250 nM T86591 CY0L2U 18442903 EC50 = 44 nM T86591 CF9BK7 18701962 EC50 = 4 nM T86591 CP8GD2 18702001 Ki = 3 nM T86591 C2GN1I 18766436 EC50 = 30 nM T86591 CYK70R 19080384 Ki = 63 nM T86591 C2C8VM 20765803 EC50 = 20 nM T86591 C3G8NO 20765805 EC50 = 20 nM T86591 CXGK50 20765807 EC50 = 14000 nM T86591 CW3G2Y 20777233 EC50 = 12 nM T86591 C59GOH 20826996 IC50 > 10000 nM T86591 C1LOC3 21054974 EC50 = 30 nM T86591 CV7UB3 21054981 EC50 = 50 nM T86591 COLV42 21054982 EC50 = 10 nM T86591 CP3RI0 21054984 EC50 = 100 nM T86591 CNW9C5 21054988 EC50 = 630 nM T86591 C5BM3O 21055003 EC50 = 190 nM T86591 CO8Z9N 21084267 EC50 = 23 nM T86591 CH51UK 21084268 EC50 = 39 nM T86591 CX2FC0 21101227 EC50 = 1800 nM T86591 C80ESD 21557355 EC50 = 28000 nM T86591 C6WHO5 21866604 EC50 = 30 nM T86591 CX48VU 21866618 EC50 = 300 nM T86591 CES61V 21866640 EC50 = 30 nM T86591 CY0TR2 21866670 EC50 = 30 nM T86591 CW70QG 21866699 EC50 = 30 nM T86591 CX2J7L 21866721 EC50 = 30 nM T86591 C3SWL4 21866734 EC50 = 3000 nM T86591 C0JZU3 21866789 EC50 = 300 nM T86591 CEMT42 21866801 EC50 = 3000 nM T86591 CMGS41 21866827 EC50 = 300 nM T86591 CV3NF2 21866832 EC50 = 3000 nM T86591 C8IH2X 21866841 EC50 = 30 nM T86591 CX05LN 21866931 EC50 = 100 nM T86591 CGHF16 21866936 EC50 = 10 nM T86591 CU0IJ4 21928218 EC50 > 10000 nM T86591 C2O4BZ 21928229 EC50 = 200 nM T86591 CEWR84 21942712 EC50 = 308 nM T86591 C48BOL 21942716 EC50 > 10000 nM T86591 CU58VO 21942721 EC50 > 10000 nM T86591 COKU53 21942723 EC50 = 220 nM T86591 CZF52L 21942731 EC50 > 10000 nM T86591 CC98SZ 21942737 EC50 = 383 nM T86591 C4T1SY 21942738 EC50 = 65 nM T86591 CAC2U8 21942751 EC50 = 327 nM T86591 CY58SO 21942772 EC50 > 10000 nM T86591 CFBM32 21942781 EC50 = 500 nM T86591 CS2U1Y 21942782 EC50 = 3890 nM T86591 CFRH71 21985914 Ki = 37 nM T86591 CI40KU 22087541 EC50 = 5 nM T86591 CN97KU 22087544 EC50 = 62 nM T86591 C6SQ5I 22087586 EC50 = 35 nM T86591 C17ZPC 22087654 EC50 = 48.6 nM T86591 CB2G3Y 22087658 EC50 = 871 nM T86591 CV0MX1 22229246 EC50 = 123 nM T86591 CU6YG1 22229249 EC50 = 297 nM T86591 C02WAZ 22229253 EC50 > 3000 nM T86591 C28MRJ 22229258 EC50 > 3000 nM T86591 C5JU1E 22229269 EC50 > 3000 nM T86591 CL01NF 22229275 EC50 > 3000 nM T86591 C4L5TH 22229292 EC50 = 643 nM T86591 C3F2OH 22229300 EC50 = 1290 nM T86591 CFA14C 22229314 EC50 = 2208 nM T86591 CSAX56 22229323 EC50 = 86 nM T86591 C8MT5I 22261152 EC50 = 81 nM T86591 CM93FV 22279993 IC50 > 10000 nM T86591 CGVR07 22280001 IC50 = 1200 nM T86591 CE3OI9 22280016 IC50 = 311 nM T86591 C1BG7A 22280047 IC50 = 3481 nM T86591 C1G2OH 22280062 IC50 = 4950 nM T86591 C14YDT 22280073 IC50 = 127.94 nM T86591 CDQ0Y6 22280103 IC50 = 790.68 nM T86591 C0VET7 22280114 IC50 = 427.56 nM T86591 C7IW1Y 22280124 IC50 = 672 nM T86591 COA0S5 22280155 IC50 = 578 nM T86591 CZS5Q3 22280173 IC50 = 3910 nM T86591 CVH3O8 22280178 IC50 > 10000 nM T86591 CE5BX0 22280187 IC50 = 4190 nM T86591 CDZB48 22280210 IC50 = 1540 nM T86591 C95ZVB 22339979 EC50 = 11 nM T86591 C7FP5O 22340076 EC50 = 7 nM T86591 CK1ZY7 22504766 IC50 = 835 nM T86591 C8CP4E 22504797 IC50 = 3840 nM T86591 C2P7OG 22504815 IC50 = 1470 nM T86591 C5YBQ0 22504835 IC50 = 1350 nM T86591 C5X6IB 22504843 IC50 = 5810 nM T86591 CDK75I 22504857 IC50 = 2380 nM T86591 CO0UC5 22504899 IC50 = 1420 nM T86591 CHD4Z0 22504917 IC50 = 311 nM T86591 CU4JP1 22610192 EC50 = 46 nM T86591 CSZ7H9 22610195 EC50 = 287 nM T86591 CE5Z8K 22610208 EC50 = 451 nM T86591 CBD72V 22708221 EC50 = 600 nM T86591 CS0HE9 22727983 EC50 = 6900 nM T86591 CE06NF 22728012 EC50 = 280 nM T86591 CG9O8Q 22928715 EC50 = 3700 nM T86591 CG23ZP 23111663 EC50 = 10000 nM T86591 CT38PB 23111732 EC50 > 10000 nM T86591 CJ5NM3 23249734 EC50 > 100000 nM T86591 CNXB90 23402689 EC50 = 1470 nM T86591 C8Z5MA 23402692 EC50 = 6 nM T86591 CU18VJ 23402759 EC50 = 311 nM T86591 CSLH35 23402760 EC50 = 120 nM T86591 CBZ85M 23402773 EC50 = 660 nM T86591 C1PBI5 23402831 EC50 > 15000 nM T86591 C14KIP 23402832 EC50 = 6150 nM T86591 C2MX7P 23529368 EC50 = 444 nM T86591 C10TAO 23553234 EC50 = 15.9 nM T86591 CEJ1S4 23628240 EC50 = 3270 nM T86591 CL6AD8 23628247 IC50 > 10000 nM T86591 CS26KY 23648476 EC50 = 2053 nM T86591 CO6EC1 23648933 EC50 = 4 nM T86591 CX8W7E 23649183 EC50 = 18 nM T86591 C18CXM 23656548 EC50 > 10000 nM T86591 C0WDH8 23657636 EC50 = 2718 nM T86591 C6CZ1W 23661590 EC50 = 10 nM T86591 CT43OQ 23661729 EC50 = 100 nM T86591 C0VKM5 23672434 EC50 = 1485 nM T86591 CZPJ84 23674509 EC50 = 1194 nM T86591 CAP8K7 23676879 EC50 > 10000 nM T86591 CY82MF 23678396 EC50 > 10000 nM T86591 C0D2NA 23683103 EC50 = 1543 nM T86591 C7W8GM 23684387 EC50 > 10000 nM T86591 C8WL4M 23684920 EC50 = 723 nM T86591 C9H4WT 23686961 EC50 > 10000 nM T86591 CF04QP 23690285 EC50 > 10000 nM T86591 C5S7GF 23703312 EC50 = 114 nM T86591 CBXC05 24424330 IC50 = 52 nM T86591 CTE1N2 24748569 EC50 > 10000 nM T86591 C56SGF 24754924 EC50 = 2824 nM T86591 CNBV74 24759099 EC50 = 8 nM T86591 CJB0Y5 24776380 EC50 = 192 nM T86591 CHE16V 24776381 EC50 > 10000 nM T86591 C5NIJ8 24776382 EC50 > 10000 nM T86591 C7EJ4W 24776383 EC50 > 10000 nM T86591 C39FEM 24776384 EC50 > 10000 nM T86591 C6WK3P 24776385 EC50 > 10000 nM T86591 COI0Q1 24776386 EC50 > 10000 nM T86591 CPI7B6 24776387 EC50 > 10000 nM T86591 CMA17V 24776388 EC50 = 6700 nM T86591 CV4CJ0 24776389 EC50 > 10000 nM T86591 CL1MV5 24776390 EC50 > 10000 nM T86591 C5J2IY 24776391 EC50 > 10000 nM T86591 CC1XW3 24776392 EC50 > 10000 nM T86591 C3RCM7 24776393 EC50 > 10000 nM T86591 C5N0IX 24776394 EC50 > 10000 nM T86591 C73QEI 24808475 EC50 > 10000 nM T86591 CLV9T5 24816384 EC50 = 1200 nM T86591 C70QHI 24828802 EC50 = 30000 nM T86591 C15NSJ 24828803 EC50 = 10000 nM T86591 CO31MA 24828805 EC50 = 14000 nM T86591 CW51RK 24828806 EC50 = 16000 nM T86591 C48SQZ 24875337 EC50 = 46.6 nM T86591 C3E7IZ 24882613 EC50 = 140 nM T86591 CP1EM0 24890166 EC50 = 6 nM T86591 C34OKV 24890167 EC50 = 74 nM T86591 C0PYD9 24890168 EC50 = 3600 nM T86591 C5Q1GX 24890333 EC50 = 53 nM T86591 C5FV9O 24890334 EC50 = 60 nM T86591 C0P4RE 24890336 EC50 = 54 nM T86591 CMU63N 24890509 EC50 = 260 nM T86591 CF57SZ 24890510 EC50 = 3.6 nM T86591 C13XCE 24890511 EC50 = 140 nM T86591 CKT23B 24890512 EC50 = 41 nM T86591 C94RLU 24890513 EC50 = 1200 nM T86591 C7LTC8 24890684 EC50 = 1400 nM T86591 C3MDU5 24890685 EC50 = 77 nM T86591 C8PD2Z 24941254 IC50 > 10000 nM T86591 C1P6WN 24949595 EC50 = 500 nM T86591 C17UHS 24949596 EC50 = 150 nM T86591 C1CG8I 24949919 EC50 = 1600 nM T86591 CX1WF4 24963031 EC50 = 623 nM T86591 CU41PY 25008799 EC50 = 7.85 nM T86591 C21QHZ 25014794 EC50 = 2800 nM T86591 CQWZ49 25032861 EC50 = 5 nM T86591 CF98EG 25071332 EC50 = 12 nM T86591 CAOE29 25104183 EC50 = 1730 nM T86591 C6WL7Z 25107241 EC50 = 1510 nM T86591 C9E4GM 25110688 EC50 = 2500 nM T86591 C8CAY3 25110733 EC50 = 240 nM T86591 CZ8AR6 25110744 EC50 = 64 nM T86591 CF3DZ4 25112371 EC50 = 12 nM T86591 CU78IR 25114869 EC50 = 2910 nM T86591 CI53RL 25114871 EC50 = 2700 nM T86591 CU1T2F 25114873 EC50 = 674 nM T86591 CDA68R 25115099 EC50 = 58800 nM T86591 C4Q1WY 25115101 EC50 = 13100 nM T86591 C0BT6Z 25115103 EC50 = 4060 nM T86591 CUW4D0 25115277 EC50 > 10000 nM T86591 CZH49S 25115278 EC50 > 10000 nM T86591 CWJ0T7 25115333 EC50 = 2950 nM T86591 CG1TV7 25115504 EC50 > 10000 nM T86591 CMK0A5 25115507 EC50 > 10000 nM T86591 C6RT7Y 25115556 EC50 = 12100 nM T86591 CF31BP 25115790 EC50 = 3990 nM T86591 CDF4J5 25115793 EC50 = 24400 nM T86591 C2H5QL 25116020 EC50 = 6780 nM T86591 CZW5M7 25116021 EC50 = 4390 nM T86591 CT93BD 25116250 EC50 = 2760 nM T86591 C2M6GN 25116484 EC50 = 37400 nM T86591 CI9SL3 25116487 EC50 = 11300 nM T86591 C4M6ZY 25116726 EC50 = 3950 nM T86591 C5F3XY 25116813 EC50 = 5900 nM T86591 C7Y4EV 25116953 EC50 = 21600 nM T86591 CHD2G4 25116956 EC50 = 3080 nM T86591 CXE3I5 25116957 EC50 = 44500 nM T86591 C57LQZ 25117176 EC50 = 3260 nM T86591 C1J5LQ 25117396 EC50 = 2270 nM T86591 C3NU1E 25132561 EC50 = 5600 nM T86591 CJ06KN 25132562 EC50 = 30400 nM T86591 C5DV8Z 25147673 EC50 = 0.072 nM T86591 CYFQ56 25147837 EC50 = 100 nM T86591 CX05GL 25147838 EC50 = 1550 nM T86591 CJAC29 25147839 EC50 = 100 nM T86591 CASK45 25147840 EC50 = 720 nM T86591 C4OVN0 25147933 EC50 = 5250 nM T86591 CXR1L0 25148011 EC50 = 2290 nM T86591 C7NXK8 25148013 EC50 = 70 nM T86591 CIN0X4 25148014 EC50 = 910 nM T86591 COS02A 25148015 EC50 = 1200 nM T86591 CX25ZB 25148016 EC50 = 910 nM T86591 C1L6RT 25148090 EC50 = 170 nM T86591 C2I9DM 25149038 EC50 = 1230 nM T86591 CC9GO5 25149124 EC50 = 1620 nM T86591 C8N3SX 25149125 EC50 = 1 nM T86591 C0Q7ZR 25149126 EC50 = 1200 nM T86591 CM4F1V 25149127 EC50 = 1290 nM T86591 CSMT48 25149129 EC50 = 1740 nM T86591 CX97GA 25164959 IC50 > 50000 nM T86591 C45WHD 25165162 IC50 > 50000 nM T86591 CZF5B0 25165359 IC50 > 50000 nM T86591 C7W3IH 25165560 IC50 > 50000 nM T86591 CZ4TN9 25165638 IC50 > 50000 nM T86591 CER49X 25165639 IC50 > 50000 nM T86591 CBPX25 25166738 IC50 > 50000 nM T86591 C3HAY5 25166740 IC50 > 50000 nM T86591 C4WNU0 25166741 IC50 > 50000 nM T86591 CPE1I4 25166743 IC50 > 50000 nM T86591 CS03PW 25166956 IC50 > 50000 nM T86591 C72AEW 25167766 IC50 = 34 nM T86591 C5RBW3 25179712 IC50 = 190 nM T86591 C64FTI 25211572 IC50 > 50000 nM T86591 CZ9H6S 25211874 EC50 = 7070 nM T86591 CT51NS 25211876 IC50 = 3162.28 nM T86591 CSWB02 25211877 IC50 = 3162.28 nM T86591 C50YNC 25243830 EC50 = 54 nM T86591 CL8A5V 25247546 EC50 = 2060 nM T86591 CR3E5T 25263358 IC50 > 10000 nM T86591 CU68GV 25263359 IC50 = 10000 nM T86591 COFY03 25263360 IC50 = 5011.87 nM T86591 CL6SG8 25263361 IC50 = 3981.07 nM T86591 CJW5Z8 25263362 IC50 = 6309.57 nM T86591 C2YU5K 25263363 IC50 = 1584.89 nM T86591 CB70OD 25263364 IC50 = 5011.87 nM T86591 CE7MW2 25263365 IC50 > 10000 nM T86591 CAM4D7 25263366 IC50 = 7943.28 nM T86591 C5KJS4 25263367 IC50 > 10000 nM T86591 CT5R1F 25263368 IC50 = 3981.07 nM T86591 CO16NL 25263369 IC50 = 5011.87 nM T86591 C6NSB5 25263370 IC50 = 10000 nM T86591 C7KPY3 25263371 IC50 = 6309.57 nM T86591 CLS1I8 25263372 IC50 = 7943.28 nM T86591 C7U4IG 25263373 IC50 = 10000 nM T86591 CJ7NW1 25263374 IC50 = 1000 nM T86591 CY09AD 25263375 IC50 = 1258.93 nM T86591 CPT2M7 25263376 IC50 = 1258.93 nM T86591 C3J6IA 25263377 IC50 = 1000 nM T86591 CJG62V 25263378 IC50 = 1995 nM T86591 CV5S1G 25263379 IC50 = 7943 nM T86591 C5QA6B 25263380 IC50 = 2511.89 nM T86591 CF49OS 25263381 IC50 = 3162.28 nM T86591 CZDA26 25263382 IC50 = 3981.07 nM T86591 CG59MP 25263383 IC50 = 1584.89 nM T86591 CD9EZ2 25263384 IC50 = 3162.28 nM T86591 C10NLX 25263385 IC50 > 10000 nM T86591 C50GAO 25263386 IC50 = 794.33 nM T86591 C8KCW3 25263387 IC50 = 3162.28 nM T86591 CJST96 25263388 IC50 = 1584.89 nM T86591 CW6U1B 25263389 EC50 > 1000 nM T86591 CKMR46 25263390 EC50 > 1000 nM T86591 CZ0CO2 25263391 EC50 > 10000 nM T86591 C3P9KJ 25263392 EC50 > 10000 nM T86591 CA8JG2 25263393 EC50 > 10000 nM T86591 C9B0PG 25263394 EC50 > 10000 nM T86591 CE35MH 25263395 EC50 > 10000 nM T86591 C3RG0W 25263396 EC50 > 10000 nM T86591 C19DVJ 25263397 EC50 > 10000 nM T86591 C3FGA6 25263398 EC50 > 10000 nM T86591 C04WDJ 25263399 EC50 > 10000 nM T86591 CHL2X3 25263400 EC50 > 10000 nM T86591 CGZL24 25263401 EC50 = 19 nM T86591 CUMZ05 25263402 EC50 = 12 nM T86591 CPO0U4 25263403 EC50 = 2.2 nM T86591 CFS9A2 25263404 EC50 = 1.3 nM T86591 CC29YB 25263405 EC50 = 3.1 nM T86591 CD9SV4 25263406 EC50 = 32 nM T86591 CJ6L2O 25263407 EC50 = 26 nM T86591 CBGE67 25263408 EC50 = 10.6 nM T86591 C08EKY 25263409 EC50 = 596 nM T86591 CH5PV6 25263410 EC50 = 12 nM T86591 C6F0WS 25263411 EC50 = 11.7 nM T86591 C78DHO 25263412 EC50 = 139 nM T86591 CBM0U5 25263413 EC50 = 10 nM T86591 C6Z2KG 42604838 EC50 = 111 nM T86591 CNU8Q0 42608446 Ki = 880 nM T86591 CX70AK 42625720 EC50 = 200 nM T86591 CW36AR 42625721 EC50 > 10000 nM T86591 CX6D9E 42625795 EC50 > 10000 nM T86591 C2TK3Z 42625796 EC50 = 30 nM T86591 CRLG64 42625797 EC50 = 1920 nM T86591 C3UKN7 42625798 EC50 = 40 nM T86591 CNE6U4 42625799 EC50 = 240 nM T86591 CVAN68 42625871 EC50 > 10000 nM T86591 CG8K1S 42625874 EC50 > 10000 nM T86591 C86XNA 42625875 EC50 > 10000 nM T86591 CW0A6E 42625952 EC50 = 130 nM T86591 C67UGQ 42625953 EC50 = 130 nM T86591 CC6YK7 42625954 EC50 = 30 nM T86591 C83VLK 42625955 EC50 = 4070 nM T86591 CC81PK 42625956 EC50 = 30 nM T86591 C04ROU 42626028 EC50 = 50 nM T86591 CI4VG0 42626029 EC50 = 120 nM T86591 CIJ3H9 42626030 EC50 = 3990 nM T86591 CUS7L8 44132498 EC50 > 10000 nM T86591 CQ83EC 44143316 Ki = 1200 nM T86591 C12XUE 44143317 Ki = 210 nM T86591 CD2VC6 44143318 Ki = 1300 nM T86591 CBOX40 44143319 Ki = 1200 nM T86591 C1GQC6 44143320 Ki = 940 nM T86591 C9FRI3 44143321 Ki = 1300 nM T86591 C3DGV4 44143322 Ki = 1300 nM T86591 C0Z8NG 44143323 Ki = 1100 nM T86591 C6GJU8 44143324 Ki = 1200 nM T86591 CK25QY 44143325 EC50 > 10000 nM T86591 C9D6TL 44143326 Ki = 960 nM T86591 C7U1JB 44143327 Ki = 1100 nM T86591 C4OBI5 44143328 Ki = 1900 nM T86591 C3ZL5T 44143329 Ki = 1700 nM T86591 CX8Z3J 44143330 Ki = 1700 nM T86591 CO72BR 44143331 Ki = 2900 nM T86591 CZ3GO9 44143332 Ki = 2000 nM T86591 C78CKO 44143333 Ki = 1700 nM T86591 CLUG09 44143334 Ki = 1000 nM T86591 C6VE7C 44143335 Ki = 1300 nM T86591 CZF3A7 44143336 Ki = 930 nM T86591 C0UKO6 44143337 Ki = 2000 nM T86591 CF2O9K 44143338 Ki = 800 nM T86591 CUG16K 44143339 Ki = 7900 nM T86591 C4MB2X 44143340 Ki = 5900 nM T86591 C7BS4Z 44143341 Ki = 5500 nM T86591 CNA0F7 44143342 Ki = 2600 nM T86591 CM3N5P 44143343 Ki = 4100 nM T86591 C5AK1N 44190592 EC50 = 4890 nM T86591 CSN2I3 44190675 EC50 = 230 nM T86591 C7VP2C 44190676 EC50 = 370 nM T86591 C2AV1K 44190762 EC50 = 320 nM T86591 C2Z9AO 44190763 EC50 = 500 nM T86591 CT2VX9 44190764 EC50 > 3000 nM T86591 C1HYW3 44190860 EC50 = 380 nM T86591 CGL02H 44190861 EC50 = 2 nM T86591 C2FIL5 44190862 EC50 = 107 nM T86591 C6MZ5G 44190863 EC50 > 3000 nM T86591 CF29RT 44241498 EC50 = 150 nM T86591 COUQ71 44241499 EC50 = 10.96 nM T86591 C1B2ED 44246273 IC50 = 676 nM T86591 CMH0A5 44246274 EC50 = 874 nM T86591 CRE63N 44246275 EC50 > 20000 nM T86591 CLM3P2 44246276 EC50 > 20000 nM T86591 CON62P 44249904 EC50 = 21 nM T86591 C98GDR 44249905 EC50 = 11 nM T86591 C5LE2G 44263416 EC50 = 1000 nM T86591 C46JLC 44263417 EC50 = 16000 nM T86591 CV24PU 44263418 EC50 > 100000 nM T86591 C63NTO 44263419 EC50 > 100000 nM T86591 CHV0U4 44263420 EC50 = 29000 nM T86591 CST49K 44263421 EC50 = 11000 nM T86591 C2IV6K 44263422 EC50 > 30000 nM T86591 CB2L5E 44263423 EC50 = 5000 nM T86591 CJ8NG4 44263424 EC50 = 25000 nM T86591 CQF3S1 44263425 EC50 > 100000 nM T86591 CK0Y7P 44263426 IC50 = 1900 nM T86591 CN8F7X 44263427 EC50 > 30000 nM T86591 CM4JU6 44263428 EC50 = 12000 nM T86591 C9ORI5 44263429 EC50 > 30000 nM T86591 C5A4HL 44273874 EC50 = 17 nM T86591 CE58NO 44273875 EC50 = 100 nM T86591 CMX75T 44273944 EC50 = 5 nM T86591 C0XNR5 44273963 EC50 = 6 nM T86591 CC06QB 44273964 EC50 = 50 nM T86591 CXOQ47 44274021 EC50 = 1 nM T86591 CBY28T 44274044 EC50 = 9 nM T86591 CNV3P0 44274047 EC50 = 20 nM T86591 CH7M5T 44274107 EC50 = 9 nM T86591 C67AKM 44316114 EC50 = 400 nM T86591 C1HKA2 44316347 EC50 = 160 nM T86591 CP3GE6 44316348 EC50 = 79 nM T86591 C27PUY 44316349 EC50 = 40 nM T86591 CJ4IP0 44316383 EC50 = 50 nM T86591 C1V6UE 44316496 EC50 = 25 nM T86591 CX1V8Q 44316506 EC50 = 79 nM T86591 CX07YR 44316521 EC50 = 13 nM T86591 C1LBQ7 44316568 EC50 = 40 nM T86591 CI19KT 44316591 EC50 = 20 nM T86591 CNG0H5 44316592 EC50 = 32 nM T86591 CDPY05 44316628 EC50 = 400 nM T86591 CXC9R4 44316629 EC50 = 790 nM T86591 C64ETY 44316824 EC50 = 40 nM T86591 CLQ0B3 44316825 EC50 = 500 nM T86591 CD2HP8 44316826 EC50 = 2000 nM T86591 C29KBV 44316844 EC50 = 240 nM T86591 CKC5F4 44316880 EC50 = 200 nM T86591 CFT53Z 44316903 EC50 = 320 nM T86591 C3E7QU 44320897 EC50 = 1096.48 nM T86591 CIY30P 44320978 EC50 = 891.25 nM T86591 C6J0GY 44321201 EC50 = 3162.28 nM T86591 CLBK38 44321284 EC50 = 300 nM T86591 C4IR1A 44321440 EC50 = 6400 nM T86591 C45WMS 44321441 EC50 = 2187.76 nM T86591 CR3T1Q 44321462 EC50 = 400 nM T86591 C9AEI4 44321463 EC50 = 2187.76 nM T86591 CRFU18 44321490 EC50 = 2000 nM T86591 CQ10AI 44321517 EC50 = 4466.84 nM T86591 CH6Z2D 44321548 EC50 = 691.83 nM T86591 C6ZK4E 44321572 EC50 = 300 nM T86591 CQ3RA9 44321573 EC50 = 691.83 nM T86591 C6HM2Z 44321655 EC50 = 5248.07 nM T86591 CH1U9W 44323732 EC50 = 14000 nM T86591 C8N7LP 44331667 EC50 = 59 nM T86591 CRG71X 44331668 EC50 = 710 nM T86591 CR9E3N 44331685 EC50 = 230 nM T86591 CTFW53 44331750 EC50 = 230 nM T86591 CRNL38 44331751 EC50 = 620 nM T86591 CQHJ92 44335944 EC50 = 6900 nM T86591 C9M2TC 44335993 Ki = 1200 nM T86591 CX1PV7 44336742 EC50 = 3380 nM T86591 CI9AN1 44337634 Ki = 225 nM T86591 CR9YS1 44337635 Ki = 57 nM T86591 CRA5F6 44337688 Ki = 18 nM T86591 CEMT31 44337693 Ki = 98 nM T86591 CZ7J0I 44337694 Ki = 12 nM T86591 C4X6LA 44337716 Ki = 28 nM T86591 CCQ67S 44337866 Ki = 28 nM T86591 CRJ87P 44338182 Ki = 293 nM T86591 CWB32K 44338195 Ki = 61 nM T86591 CA36CR 44339522 EC50 = 10 nM T86591 CV3R2S 44339547 EC50 = 4200 nM T86591 CZ25OL 44344272 EC50 = 90 nM T86591 C9C8FN 44344313 EC50 = 170 nM T86591 CWD8B7 44344585 EC50 = 140 nM T86591 CMC41U 44345158 Ki = 21000 nM T86591 C4MTA7 44345159 Ki > 100000 nM T86591 CR0GI8 44345164 Ki > 100000 nM T86591 CR7EX2 44345170 Ki > 100000 nM T86591 CX2I7F 44345171 Ki = 67000 nM T86591 CH9F6O 44345180 Ki > 100000 nM T86591 CXY46J 44345202 EC50 = 5000 nM T86591 CU7F4O 44345203 EC50 = 3800 nM T86591 CC3FJ0 44345204 Ki > 100000 nM T86591 CMR75E 44345354 Ki > 100000 nM T86591 C5WY9X 44345355 Ki > 100000 nM T86591 CANH09 44345363 EC50 = 12000 nM T86591 CPHO86 44345406 EC50 = 10000 nM T86591 C2FGP1 44345407 EC50 = 2500 nM T86591 C2BKP7 44345432 Ki > 100000 nM T86591 CY7O8G 44345843 EC50 = 1000 nM T86591 C1B2CN 44345903 EC50 = 290 nM T86591 CU6HZ2 44345963 EC50 = 360 nM T86591 C0CS9D 44348875 EC50 = 150 nM T86591 C5IE3N 44364876 Ki = 1412.54 nM T86591 CS3C7W 44365532 EC50 = 220 nM T86591 CM1X4H 44379496 EC50 = 12400 nM T86591 CZ5BG6 44383664 Ki = 46 nM T86591 CK9PD5 44383828 EC50 = 4 nM T86591 CIVC76 44383831 EC50 = 53 nM T86591 CMB3S2 44383889 Ki = 7.6 nM T86591 C5ND3Y 44384224 Ki = 920 nM T86591 CW9LD2 44384226 EC50 = 2 nM T86591 CPY0K6 44384403 EC50 = 33 nM T86591 CD4KM5 44384407 Ki = 50 nM T86591 C53DOZ 44384408 Ki > 33330 nM T86591 CTJD81 44384415 Ki = 76 nM T86591 CKDS82 44384419 EC50 = 2 nM T86591 CA7YK9 44384460 EC50 = 13 nM T86591 C4W7VN 44384466 Ki = 86 nM T86591 C46RVE 44384539 Ki = 133 nM T86591 C6PIU9 44384589 EC50 = 10 nM T86591 C4R6EW 44384639 EC50 = 2 nM T86591 CM8AE6 44385177 Ki = 489 nM T86591 C2FQX7 44385248 Ki = 5.2 nM T86591 CFM56P 44385352 Ki = 329 nM T86591 CE47ZL 44385396 EC50 = 92 nM T86591 C6H0OL 44385399 Ki = 53 nM T86591 CY2O5S 44385405 Ki = 11 nM T86591 CH9UP4 44385406 EC50 = 3 nM T86591 CRWI98 44386508 EC50 = 3 nM T86591 CDN54E 44388167 IC50 > 15000 nM T86591 C50FPR 44388210 EC50 = 130 nM T86591 C5DNU7 44388563 EC50 = 300 nM T86591 C51XZF 44388650 IC50 = 3900 nM T86591 C8E1NU 44388684 IC50 > 15000 nM T86591 CA1XK7 44388810 EC50 = 220 nM T86591 CU1Y8L 44388819 EC50 = 240 nM T86591 CU71OL 44388848 EC50 = 420 nM T86591 C28TPK 44388866 EC50 = 23 nM T86591 CMQ25R 44388882 EC50 = 40 nM T86591 CQ6Z4Y 44388907 EC50 = 140 nM T86591 CBV25F 44388914 EC50 = 4 nM T86591 C0EH5G 44388966 IC50 = 1650 nM T86591 CF7L8V 44388968 EC50 = 1000 nM T86591 C5V0PS 44389085 IC50 = 1640 nM T86591 C0S6QK 44389098 IC50 = 2750 nM T86591 C6GF3L 44389191 EC50 = 61 nM T86591 CGP9F0 44389687 EC50 = 14000 nM T86591 C1UGI7 44389733 EC50 = 300 nM T86591 C5Y3AZ 44389800 EC50 = 15000 nM T86591 COXA71 44389801 EC50 = 1600 nM T86591 CX5A2Z 44389847 EC50 = 1000 nM T86591 C78VSM 44392315 IC50 = 309.03 nM T86591 C83DZJ 44396236 EC50 = 10 nM T86591 C60YCL 44404190 IC50 = 4400 nM T86591 C21HNW 44404248 EC50 > 10000 nM T86591 CD79BV 44404256 EC50 > 10000 nM T86591 CMQI41 44404263 EC50 = 262 nM T86591 C6G1EF 44404267 EC50 = 1454 nM T86591 CGX5M8 44404271 EC50 = 1531 nM T86591 CICB09 44404275 EC50 > 10000 nM T86591 CGD96V 44404636 IC50 > 15000 nM T86591 C5F9ZX 44404637 IC50 > 15000 nM T86591 CQ9V3L 44404648 IC50 > 15000 nM T86591 CL3OB9 44404649 IC50 > 50000 nM T86591 C6EIY9 44404654 IC50 > 50000 nM T86591 CR59YU 44404675 IC50 = 3577 nM T86591 CZ53YS 44404680 IC50 > 50000 nM T86591 CUX13J 44404681 IC50 > 50000 nM T86591 C6D7SO 44404685 IC50 > 50000 nM T86591 CUX92K 44404686 IC50 = 3197 nM T86591 C4TQ6X 44404690 IC50 > 15000 nM T86591 CY35ZW 44404691 IC50 > 15000 nM T86591 C8RPC4 44404696 IC50 > 50000 nM T86591 C7Z5ST 44404700 IC50 > 15000 nM T86591 C5IUA7 44404701 IC50 > 15000 nM T86591 CS8NO5 44404703 IC50 > 15000 nM T86591 CL30JV 44404704 IC50 > 15000 nM T86591 C7GNI4 44404708 IC50 > 15000 nM T86591 C48RBM 44404714 IC50 > 4482 nM T86591 CJH5X6 44404715 IC50 > 15000 nM T86591 CHNT04 44404717 IC50 > 50000 nM T86591 C7ZSM1 44404718 IC50 = 6271 nM T86591 CT15BE 44404723 IC50 = 4154 nM T86591 C3UB2D 44404727 IC50 = 9024 nM T86591 C5GZP7 44404728 IC50 = 11475 nM T86591 COI8L9 44404729 IC50 > 15000 nM T86591 CM96VZ 44404734 IC50 > 50000 nM T86591 CP7U3J 44404735 IC50 > 50000 nM T86591 C7IJ5H 44405121 EC50 = 1209 nM T86591 CFZB63 44406104 EC50 = 204 nM T86591 CDAF49 44406106 EC50 = 637 nM T86591 CDA3Z9 44406117 EC50 = 745 nM T86591 CJ7F5L 44406154 EC50 = 718 nM T86591 CC0Y3J 44406172 EC50 = 559 nM T86591 CS06AB 44406180 EC50 = 1170 nM T86591 CA1XV3 44406204 EC50 = 75 nM T86591 CB1X2D 44406205 EC50 = 1130 nM T86591 C7AD9N 44406236 EC50 = 523 nM T86591 CB0E4H 44406258 EC50 > 10000 nM T86591 CI47RY 44406262 EC50 = 1220 nM T86591 CSO0P7 44406263 EC50 = 1000 nM T86591 C95DYP 44406265 EC50 = 5480 nM T86591 C2XDJ1 44406266 EC50 = 29 nM T86591 C7K6HJ 44406267 EC50 = 670 nM T86591 C3I0MQ 44406283 EC50 = 7260 nM T86591 CK4Z7J 44406288 EC50 = 232 nM T86591 CXY5J2 44406292 EC50 = 3280 nM T86591 CUW97K 44406303 EC50 > 10000 nM T86591 C6KL7U 44406304 EC50 > 10000 nM T86591 CA91XP 44406318 EC50 > 10000 nM T86591 CPN2F1 44406331 EC50 = 6000 nM T86591 C13MXB 44406336 EC50 = 5790 nM T86591 C9GNW2 44406340 EC50 = 979 nM T86591 CT4Z8O 44406341 EC50 = 1040 nM T86591 CB6S1C 44406344 EC50 = 232 nM T86591 C0WAS9 44406345 EC50 > 10000 nM T86591 CRY47S 44406364 EC50 > 10000 nM T86591 C5U1OQ 44406365 EC50 > 10000 nM T86591 C3KIO7 44406367 EC50 = 670 nM T86591 CQ20JM 44406375 EC50 = 868 nM T86591 CK10VQ 44406381 EC50 = 94 nM T86591 C1WPX7 44406411 EC50 = 48 nM T86591 C4IBL1 44406437 EC50 = 795 nM T86591 CV5L8T 44406441 EC50 > 10000 nM T86591 C7R5NB 44406455 EC50 = 63 nM T86591 C2Z7XC 44406472 EC50 > 10000 nM T86591 CKA1Z0 44406477 EC50 = 62 nM T86591 C1OFD9 44406482 EC50 = 57 nM T86591 C4IOC7 44406528 EC50 = 827 nM T86591 CW70MB 44406532 EC50 = 26 nM T86591 C0Y4EZ 44406533 EC50 = 350 nM T86591 CDX97W 44407180 EC50 = 150 nM T86591 CU24FD 44407220 EC50 = 20 nM T86591 CJO4I9 44407221 EC50 = 25 nM T86591 C7X4UM 44407224 EC50 = 250 nM T86591 C71EIZ 44409030 IC50 = 537 nM T86591 CD7W9V 44409035 EC50 = 44 nM T86591 C3I7OD 44409044 EC50 = 20 nM T86591 C82CKD 44409063 IC50 = 157 nM T86591 CTA6G7 44409088 EC50 = 51 nM T86591 CWGR81 44409098 EC50 = 2.1 nM T86591 C29VWO 44409126 EC50 = 3 nM T86591 C6TRF5 44409127 EC50 = 20 nM T86591 CJ8A6M 44409131 IC50 = 41.98 nM T86591 C6Y1XC 44409170 IC50 = 675 nM T86591 CEBA60 44409171 IC50 = 208 nM T86591 CB02UG 44409181 EC50 = 35 nM T86591 C1BE3K 44409183 IC50 = 125 nM T86591 CTE3C9 44409198 EC50 = 62 nM T86591 CK45XW 44409199 EC50 = 21 nM T86591 C90PQA 44409212 EC50 = 10 nM T86591 CU3Z9B 44409213 IC50 = 6090 nM T86591 C7FMA5 44409249 EC50 = 1 nM T86591 C92WDV 44409251 EC50 = 7.8 nM T86591 CRV6M9 44409273 EC50 = 11.4 nM T86591 C51XIC 44409274 EC50 = 2.9 nM T86591 CAN69Y 44409279 EC50 < 1 nM T86591 CH5B7Q 44409318 IC50 = 156 nM T86591 CZI2T9 44409319 EC50 = 454 nM T86591 C17ZLP 44409323 IC50 = 262 nM T86591 C76RXA 44409375 EC50 = 27.5 nM T86591 C3ODA1 44409427 EC50 = 2.5 nM T86591 C5LH3D 44409429 EC50 = 2.7 nM T86591 C9D7YM 44409430 EC50 = 15 nM T86591 C3F9ZO 44409437 EC50 = 10 nM T86591 CU30EB 44411547 EC50 > 10000 nM T86591 CYER28 44411548 EC50 > 10000 nM T86591 CBYE57 44411557 EC50 > 10000 nM T86591 CWR6V3 44411558 EC50 > 10000 nM T86591 C5IWC6 44411561 EC50 > 10000 nM T86591 C8G1HJ 44411562 EC50 > 10000 nM T86591 CNO49B 44411563 EC50 > 10000 nM T86591 C25NTU 44411565 EC50 > 10000 nM T86591 C3G2CA 44411571 EC50 > 10000 nM T86591 C4W6DO 44411577 EC50 > 10000 nM T86591 CFB63G 44411578 EC50 > 10000 nM T86591 CM0RU6 44411581 EC50 > 10000 nM T86591 COB80S 44411616 EC50 > 10000 nM T86591 C4C9LD 44411618 EC50 > 10000 nM T86591 CY8K9S 44411630 EC50 > 10000 nM T86591 CNL81R 44411653 IC50 = 230 nM T86591 CW3AV8 44411661 IC50 = 19 nM T86591 C5P4BM 44411708 EC50 > 10000 nM T86591 C5AR4E 44411737 EC50 > 10000 nM T86591 C06BPM 44411740 EC50 > 10000 nM T86591 C2G1LB 44411741 EC50 > 10000 nM T86591 CQL2Z4 44411767 EC50 > 10000 nM T86591 C2KCO7 44411772 EC50 > 10000 nM T86591 C4MAN2 44411789 IC50 = 2600 nM T86591 C4U2SJ 44411842 IC50 = 309.74 nM T86591 CJF9L1 44411843 IC50 = 16 nM T86591 CV3N5O 44411918 EC50 > 10000 nM T86591 CFU5X3 44411943 EC50 = 1640 nM T86591 CP1AZ6 44411945 EC50 = 730 nM T86591 C70NKQ 44411946 EC50 > 10000 nM T86591 C71ZSM 44411968 EC50 > 10000 nM T86591 CX6DN0 44411977 IC50 = 1499.68 nM T86591 CBVJ21 44412006 IC50 = 140 nM T86591 C8DPK5 44412188 IC50 = 599.79 nM T86591 CPK6G2 44412195 IC50 = 870 nM T86591 C1GH3B 44414891 EC50 > 10000 nM T86591 CU8NQ5 44414900 EC50 > 10000 nM T86591 CKM0I8 44414901 EC50 > 10000 nM T86591 C7LCH5 44414917 EC50 = 7110 nM T86591 CBQ62J 44414926 EC50 > 10000 nM T86591 C07VTH 44414927 EC50 = 1670 nM T86591 C1ETO8 44414955 EC50 > 10000 nM T86591 CV8IA5 44414956 EC50 > 10000 nM T86591 CTK8Z0 44414962 EC50 > 10000 nM T86591 C1G4OC 44414967 EC50 > 10000 nM T86591 C64UOB 44414968 EC50 > 10000 nM T86591 CLO83A 44414991 EC50 = 220 nM T86591 C23ARN 44415004 EC50 = 340 nM T86591 C0TI2L 44415602 EC50 = 1010 nM T86591 C4ZDC7 44415616 EC50 = 103 nM T86591 C04EOY 44415664 EC50 = 1068 nM T86591 C1UO6R 44415696 EC50 = 8391 nM T86591 C6C0YB 44415715 EC50 = 1401 nM T86591 C4OS6D 44418903 EC50 = 524 nM T86591 C9NB7J 44419009 EC50 = 120 nM T86591 C97QXT 44419013 EC50 = 1890 nM T86591 CP0F9T 44419760 EC50 = 65 nM T86591 CBZ5D8 44419765 EC50 = 426 nM T86591 CC6U1K 44419769 EC50 = 430 nM T86591 C17UJG 44419770 EC50 = 9400 nM T86591 C2A5CS 44419772 EC50 = 31 nM T86591 C0J5VZ 44419773 EC50 = 534 nM T86591 CCA53N 44419776 EC50 = 33 nM T86591 CF6E9L 44419778 EC50 = 13 nM T86591 CT8CU5 44419780 EC50 = 4670 nM T86591 CWK6C9 44419783 EC50 = 1230 nM T86591 CL74CP 44419785 EC50 = 6150 nM T86591 C6Z9KE 44419786 EC50 = 238 nM T86591 CUQJ29 44419790 EC50 = 8300 nM T86591 C3K6RF 44419795 EC50 = 32 nM T86591 C39JPK 44419805 EC50 = 1840 nM T86591 CM2YG0 44419807 Ki = 1800 nM T86591 C8E6CZ 44419808 EC50 = 23 nM T86591 C2ABF5 44419809 EC50 = 134 nM T86591 C7XB3Q 44419814 EC50 = 10 nM T86591 CKOR70 44419819 EC50 = 11 nM T86591 C03BNV 44419822 EC50 = 287 nM T86591 CNX3V9 44419827 EC50 = 150 nM T86591 CN62LT 44419828 EC50 = 770 nM T86591 CT8OY2 44419830 EC50 = 8 nM T86591 CY60PA 44419884 Ki = 840 nM T86591 CH8RG7 44419890 EC50 = 437 nM T86591 CP8OT7 44419891 EC50 = 48 nM T86591 C7XY6Z 44419898 Ki = 1200 nM T86591 C9FXY7 44419906 EC50 = 867 nM T86591 CY2QX8 44419911 Ki = 7300 nM T86591 CC7PF3 44419918 EC50 > 10000 nM T86591 CCI9O8 44419924 EC50 = 100 nM T86591 C4HR6P 44420473 IC50 > 10000 nM T86591 CL9N8S 44420479 EC50 = 2801 nM T86591 C5IQ7K 44420484 EC50 = 2940 nM T86591 CZ67XE 44420485 EC50 = 198 nM T86591 C5QOU1 44420506 EC50 = 35 nM T86591 CBWX49 44420565 EC50 = 2780 nM T86591 C72TSL 44420566 EC50 = 1715 nM T86591 CH1R7M 44420600 EC50 = 101 nM T86591 CL86VI 44424582 EC50 = 12 nM T86591 CV8X0N 44424583 EC50 = 520 nM T86591 C4QN7D 44424584 EC50 > 10000 nM T86591 CK89CE 44424585 EC50 = 7.9 nM T86591 CNS39L 44424586 EC50 = 41 nM T86591 CGCJ17 44424587 EC50 = 280 nM T86591 C6LXQ5 44424588 EC50 = 620 nM T86591 CBZ1C3 44424589 EC50 = 210 nM T86591 CBZU45 44424590 EC50 = 19 nM T86591 CC32AV 44424591 EC50 = 70 nM T86591 CQ1KL3 44424592 EC50 = 230 nM T86591 CG1CE6 44424593 EC50 = 29 nM T86591 CL2K0C 44424594 EC50 = 140 nM T86591 CSGM27 44424595 EC50 = 820 nM T86591 C30EJO 44425850 EC50 > 1000 nM T86591 CQ9RH6 44425851 EC50 > 1000 nM T86591 CH13TY 44425852 EC50 > 1000 nM T86591 CGE39L 44425853 EC50 > 1000 nM T86591 CX39CR 44425854 EC50 > 1000 nM T86591 CBJU72 44425855 EC50 > 1000 nM T86591 C3QLV7 44425856 EC50 > 1000 nM T86591 CZ3X6Y 44425859 EC50 > 1000 nM T86591 CN8A9Y 44425862 EC50 > 1000 nM T86591 CP7JN9 44425864 EC50 > 1000 nM T86591 CP6SO9 44425869 EC50 > 1000 nM T86591 CDVH71 44425872 EC50 > 1000 nM T86591 CI0Q3G 44431866 EC50 = 260 nM T86591 CYIK84 44431867 EC50 = 70 nM T86591 C6C0VT 44431868 EC50 = 5250 nM T86591 COF38E 44431869 EC50 = 2770 nM T86591 C8QW9M 44431873 EC50 = 880 nM T86591 C9MRU3 44431876 EC50 = 380 nM T86591 CX5QL8 44431880 EC50 = 20400 nM T86591 CC81BQ 44431882 EC50 = 3940 nM T86591 CVHO05 44431883 EC50 = 7260 nM T86591 CZ9RU5 44431884 EC50 = 10700 nM T86591 C05BKW 44431885 EC50 = 6050 nM T86591 C86NSF 44431886 EC50 = 1470 nM T86591 CAPN49 44431887 EC50 = 6210 nM T86591 CV6H9Z 44432125 IC50 = 3110 nM T86591 CP0VK2 44432126 IC50 = 3670 nM T86591 CORG53 44432127 IC50 > 10000 nM T86591 C7L1WG 44432395 IC50 = 679 nM T86591 C06KRB 44432398 IC50 = 682.34 nM T86591 CWDS06 44432399 IC50 = 1040 nM T86591 C9YZ1I 44432400 IC50 = 7860 nM T86591 CK6PU9 44432401 IC50 = 4680 nM T86591 CSF09X 44432402 IC50 = 963 nM T86591 CE51LN 44432403 IC50 = 229.09 nM T86591 CDV5O8 44432404 IC50 > 10000 nM T86591 CN7KJ9 44432405 IC50 = 2500.35 nM T86591 CMO9I5 44432406 IC50 = 2380 nM T86591 CA7OU6 44432407 IC50 = 550 nM T86591 C12ANM 44432408 IC50 > 10000 nM T86591 CQ1W3L 44432409 IC50 = 179 nM T86591 C8AQ3I 44432410 IC50 = 562 nM T86591 CJ7GY1 44432411 IC50 = 172 nM T86591 CI45BS 44432832 EC50 > 10000 nM T86591 CRPF69 44432835 EC50 > 10000 nM T86591 CXR1O2 44432841 EC50 > 10000 nM T86591 CEN1Z6 44432844 EC50 > 10000 nM T86591 C1RN4F 44432845 EC50 > 10000 nM T86591 CA1GL7 44432846 EC50 > 10000 nM T86591 CLZF68 44432847 EC50 > 10000 nM T86591 C0BO8H 44432848 EC50 > 10000 nM T86591 C5C4HV 44432849 EC50 > 10000 nM T86591 C2D5YP 44432852 EC50 > 10000 nM T86591 CBC74Q 44432853 EC50 = 5800 nM T86591 C1A9NX 44432854 EC50 > 10000 nM T86591 CF3L8X 44432855 EC50 = 4100 nM T86591 C9ETG7 44432856 EC50 > 10000 nM T86591 CKTE10 44432857 EC50 = 14000 nM T86591 CWF49O 44434337 EC50 = 1253 nM T86591 C53YEQ 44434338 EC50 = 828 nM T86591 C74NKE 44434339 EC50 = 836 nM T86591 C43PNF 44434340 EC50 = 466 nM T86591 CGD7Q8 44434341 EC50 = 590 nM T86591 CQP74N 44434342 IC50 = 10303.86 nM T86591 CVWA23 44434343 EC50 = 706 nM T86591 C0VAZ9 44434344 EC50 = 329 nM T86591 C5WY9B 44434345 EC50 = 1042 nM T86591 CM4K1D 44434346 EC50 = 2205 nM T86591 CKI70B 44434347 EC50 = 420 nM T86591 CH5JP2 44434348 EC50 = 1504 nM T86591 CQW7J6 44434349 EC50 = 2727 nM T86591 CS31PG 44434350 IC50 = 187.93 nM T86591 CERT39 44434351 IC50 = 331 nM T86591 C4B8VJ 44434352 IC50 = 727.78 nM T86591 CM8VY6 44434353 IC50 = 384 nM T86591 C9IG2C 44434354 EC50 = 2997 nM T86591 C4SMI1 44434355 EC50 = 2459 nM T86591 C3O2BF 44434356 EC50 = 588 nM T86591 CRBM37 44434357 EC50 = 2770 nM T86591 CL2H8U 44434358 EC50 = 2404 nM T86591 CB5U3S 44434359 EC50 = 1887 nM T86591 C4K0FY 44434360 EC50 = 2735 nM T86591 CIA86O 44434361 EC50 = 558 nM T86591 C2VG9W 44434362 IC50 = 9332.54 nM T86591 CL5AH3 44439623 IC50 = 5950 nM T86591 CF01IC 44439624 EC50 = 2690 nM T86591 C64AHD 44439625 EC50 = 2800 nM T86591 CIW8B5 44439626 EC50 = 2900 nM T86591 CL1XI5 44439632 EC50 = 2810 nM T86591 CM6Q0Y 44439633 EC50 = 2340 nM T86591 CBQ3V5 44439710 EC50 = 6610 nM T86591 CUF6W1 44439711 EC50 = 1150 nM T86591 CB1RK5 44439712 EC50 = 1390 nM T86591 CQW59J 44439713 EC50 = 6550 nM T86591 CUJP69 44439715 EC50 = 2120 nM T86591 CK14PR 44439716 EC50 = 1130 nM T86591 CL9U1M 44439718 EC50 = 4390 nM T86591 C5O8ZX 44439719 EC50 = 3540 nM T86591 CBM0E7 44439721 EC50 = 2370 nM T86591 CR2VY5 44439724 EC50 = 565 nM T86591 CO7CV3 44439725 EC50 = 425 nM T86591 C2RNS5 44439726 EC50 = 120 nM T86591 CVS0Q5 44439729 EC50 = 920 nM T86591 CU0JA6 44439730 EC50 = 807 nM T86591 C1JAZ3 44440776 EC50 = 3 nM T86591 CYOD04 44440777 EC50 = 5 nM T86591 CIR27Y 44440779 EC50 = 2 nM T86591 CG43HK 44440780 EC50 = 23 nM T86591 CNI45S 44440781 EC50 = 100 nM T86591 CQ25AW 44440782 EC50 = 5 nM T86591 CWO5C2 44440783 EC50 = 160 nM T86591 C3-OCT 44440785 EC50 = 180 nM T86591 C6TMR4 44440786 EC50 = 7 nM T86591 C03TVK 44440787 EC50 = 24 nM T86591 C1V0CH 44440788 EC50 = 120 nM T86591 C4NDM7 44440789 EC50 = 1 nM T86591 COI23R 44440790 EC50 = 1 nM T86591 C8TOE9 44440791 EC50 = 1 nM T86591 C4BQ1C 44440792 EC50 = 11 nM T86591 CDZ45N 44440795 EC50 = 2 nM T86591 CA7G3R 44440797 EC50 = 260 nM T86591 C1PQ7V 44440800 EC50 = 2 nM T86591 CX3P1C 44440804 EC50 = 130 nM T86591 C62VTF 44440805 EC50 = 3 nM T86591 CWDC32 44440806 EC50 = 20 nM T86591 C9F4ME 44440929 EC50 = 4460 nM T86591 CUJ8X0 44441213 EC50 = 300 nM T86591 CRWN48 44441214 EC50 = 60 nM T86591 CV6RK5 44441215 EC50 = 20 nM T86591 CQ23GJ 44441216 EC50 = 4 nM T86591 CX5M7Q 44441220 EC50 = 50 nM T86591 CY74RZ 44441221 EC50 = 500 nM T86591 C3AS9D 44441223 EC50 = 90 nM T86591 CBY9C7 44441224 EC50 = 30 nM T86591 CEP16Z 44441344 EC50 = 20 nM T86591 CTE95F 44441446 EC50 = 44 nM T86591 C8YB9P 44441447 EC50 = 47 nM T86591 C7M2GD 44441451 EC50 = 324 nM T86591 CZ41WB 44441453 EC50 = 313 nM T86591 C3FJM9 44441455 EC50 = 197 nM T86591 CY64MC 44441459 EC50 = 180 nM T86591 CS9OP6 44441462 EC50 = 726 nM T86591 C0RAC7 44441463 EC50 = 128 nM T86591 CBTE20 44441464 EC50 = 4 nM T86591 C06SRV 44441466 EC50 = 189 nM T86591 C9TRS0 44441467 EC50 = 21 nM T86591 CM1HQ6 44441469 IC50 = 90 nM T86591 C19DQE 44442440 EC50 = 2190 nM T86591 C2YD9E 44442441 EC50 = 2464 nM T86591 C1APG0 44442442 EC50 = 798 nM T86591 C6RVT7 44442443 EC50 = 1890 nM T86591 CAW91Q 44442444 EC50 = 78 nM T86591 CT68PM 44442445 EC50 = 546 nM T86591 C0IGW2 44442446 EC50 = 300 nM T86591 C8A6SM 44442447 EC50 = 1690 nM T86591 CPFJ29 44442448 EC50 = 504 nM T86591 CF3D6P 44442449 EC50 = 1152 nM T86591 CMQ17O 44442450 EC50 = 1188 nM T86591 CL4K7X 44442451 EC50 = 10000 nM T86591 CGCN21 44442452 EC50 = 594 nM T86591 CM1PL8 44442453 EC50 = 6960 nM T86591 CORC37 44442454 EC50 = 2270 nM T86591 C13HNY 44442455 EC50 = 6530 nM T86591 C16NTG 44442456 EC50 = 10000 nM T86591 C31ZGW 44442457 EC50 = 10000 nM T86591 CLJ21W 44442458 EC50 = 10000 nM T86591 CN14PT 44442459 EC50 = 6790 nM T86591 CY1BJ8 44442460 EC50 = 10000 nM T86591 C9EB3R 44442461 EC50 = 7940 nM T86591 CO3GE5 44442462 EC50 = 10000 nM T86591 CJ14GS 44442463 EC50 = 10000 nM T86591 CEQB08 44442464 EC50 = 10000 nM T86591 CYZA32 44442465 EC50 = 10000 nM T86591 C3LA4I 44442466 EC50 = 10000 nM T86591 C5VRE4 44442467 EC50 = 10000 nM T86591 CYUR21 44442468 EC50 = 10000 nM T86591 CM6IW4 44442469 EC50 = 10000 nM T86591 CORA57 44442470 EC50 = 10000 nM T86591 CA7MO3 44442471 EC50 = 10000 nM T86591 CU0H8W 44442472 EC50 = 1020 nM T86591 C6M0JQ 44442473 EC50 = 2530 nM T86591 CH8SN0 44442474 EC50 = 10000 nM T86591 C37QUO 44442475 EC50 = 10000 nM T86591 C31WIL 44446245 EC50 = 450 nM T86591 CI64WZ 44446247 EC50 > 10000 nM T86591 C6XIU3 44446250 EC50 > 10000 nM T86591 CHY27Q 44446252 EC50 > 10000 nM T86591 CE1S5F 44446255 EC50 = 60 nM T86591 C9OGX2 44446257 EC50 = 1000 nM T86591 CI49YJ 44446258 EC50 = 50 nM T86591 CSH1U8 44446260 EC50 = 320 nM T86591 C7YSZ5 44446262 EC50 = 0.3 nM T86591 C9GMW7 44446263 EC50 = 3 nM T86591 CIR02A 44446264 EC50 = 80 nM T86591 CD9O0L 44446265 EC50 = 60 nM T86591 CF7Z3H 44446266 EC50 = 5000 nM T86591 CB8L4Q 44446268 EC50 = 70 nM T86591 C2EUO0 44446269 EC50 = 20 nM T86591 CM4L3Y 44446271 EC50 = 1000 nM T86591 C8OCS0 44446272 EC50 = 360 nM T86591 CC5TR9 44446274 EC50 = 3000 nM T86591 C21UBL 44446281 EC50 = 80 nM T86591 C4VMW1 44446282 EC50 = 2800 nM T86591 CV0N6W 44446283 EC50 = 80 nM T86591 C6QSV8 44446284 EC50 = 6000 nM T86591 C3T2VM 44447156 EC50 = 152 nM T86591 CEJV01 44447159 EC50 = 19 nM T86591 CI97LH 44447160 EC50 = 14 nM T86591 CUL81F 44447162 EC50 = 11 nM T86591 C4QYL8 44447163 EC50 = 65 nM T86591 C5TKE9 44448345 IC50 = 3740 nM T86591 CI6HR5 44448403 EC50 = 1940 nM T86591 CTH06F 44448484 IC50 > 15000 nM T86591 C3DO6H 44448487 IC50 > 15000 nM T86591 C4KSB3 44448593 EC50 > 25000 nM T86591 CE29ID 44448632 IC50 > 15000 nM T86591 CE09DJ 44448767 EC50 = 1120 nM T86591 C1NX8Y 44448801 EC50 = 4650 nM T86591 CRK9D8 44449001 EC50 = 8 nM T86591 C4HAK6 44449024 EC50 = 24 nM T86591 CW3BX7 44449049 EC50 = 180 nM T86591 CR94MO 44449074 EC50 > 3500 nM T86591 CC90BY 44449076 EC50 = 644 nM T86591 C8DS6T 44449100 EC50 = 1290 nM T86591 CX0FP8 44449101 EC50 = 490 nM T86591 CF8U1H 44449125 EC50 = 18 nM T86591 CD1Q7S 44449127 EC50 = 1070 nM T86591 CW9YO3 44449128 EC50 > 7500 nM T86591 C1E5UC 44449161 EC50 = 263 nM T86591 C9P7JK 44449163 EC50 = 257 nM T86591 CP54JF 44449192 EC50 = 3860 nM T86591 CR1W3G 44449220 EC50 > 7500 nM T86591 C85TKY 44451190 EC50 = 155 nM T86591 CUM0J1 44453644 EC50 > 7500 nM T86591 CX46EF 44453670 EC50 > 7500 nM T86591 CXPD58 44453913 EC50 = 970 nM T86591 C6C8NI 44453940 EC50 = 90 nM T86591 C9YUM3 44453941 EC50 = 5400 nM T86591 CVI8M4 44453962 EC50 = 230 nM T86591 C63TBK 44453988 EC50 = 11 nM T86591 C5AEL6 44454012 EC50 = 140 nM T86591 C7PA9S 44454244 EC50 = 500 nM T86591 C84FIQ 44454301 EC50 = 28 nM T86591 CIE06L 44454336 EC50 = 37 nM T86591 CP8OE3 44454364 EC50 = 100 nM T86591 CA84BK 44454366 EC50 = 1700 nM T86591 CLUF89 44458859 EC50 = 1600 nM T86591 CC86GW 44458943 EC50 = 1300 nM T86591 CR5SI0 44476535 EC50 > 10000 nM T86591 C2A3XQ 44478369 EC50 = 2500 nM T86591 CZ0U2L 44478370 EC50 = 45800 nM T86591 CNE9F3 44478371 EC50 = 45800 nM T86591 C4IX8S 44478372 EC50 = 36100 nM T86591 C8S6MB 44478373 EC50 = 9300 nM T86591 CWZ8Q0 44478374 EC50 = 33300 nM T86591 CL4V1X 44478375 EC50 = 9800 nM T86591 C8QY4B 44478642 EC50 = 55900 nM T86591 CM40CQ 44478643 EC50 = 57300 nM T86591 C3LXZ1 44479180 EC50 = 46300 nM T86591 CANO48 44479182 EC50 = 38900 nM T86591 CO1IH9 44479184 EC50 = 69300 nM T86591 CD2W6Z 44479185 EC50 = 62500 nM T86591 CZU79G 44479187 EC50 = 84300 nM T86591 C2YX5E 44479188 EC50 = 9300 nM T86591 CQIG01 44479438 EC50 = 14800 nM T86591 CE0F7W 44479442 EC50 = 73500 nM T86591 CE4D5N 44479443 EC50 = 1900 nM T86591 C0ZKT3 44480200 EC50 = 330 nM T86591 C2JMV3 44480201 EC50 = 488 nM T86591 C42PIO 44480202 EC50 = 3600 nM T86591 CXVI34 44480461 EC50 = 1360 nM T86591 C1Y5EX 44480465 EC50 = 2400 nM T86591 CBJ58K 44480717 EC50 = 160 nM T86591 C89YIZ 44480973 EC50 = 60 nM T86591 CJ6O7D 44481226 EC50 = 600 nM T86591 CY69AT 44481227 EC50 = 310 nM T86591 C39MBW 44481228 EC50 = 1400 nM T86591 C60RWZ 44481229 EC50 = 1750 nM T86591 CEM86S 44481230 EC50 = 720 nM T86591 CO06ZF 44481496 EC50 = 1800 nM T86591 CM4Z1D 44515004 EC50 = 19000 nM T86591 CI4A7H 44515005 IC50 = 2480 nM T86591 CU10OJ 44515008 IC50 = 3330 nM T86591 CPW0S4 44561816 IC50 > 50000 nM T86591 C9L3VY 44561817 IC50 > 50000 nM T86591 C08NKI 44561969 IC50 > 50000 nM T86591 CS48WU 44562841 EC50 > 25000 nM T86591 C94SYK 44562842 EC50 > 25000 nM T86591 CG13BO 44564813 EC50 > 15000 nM T86591 CVN24W 44564853 EC50 = 11 nM T86591 CG1Q3X 44564854 EC50 = 648 nM T86591 CVZA94 44564855 EC50 = 126 nM T86591 CUA0F7 44564899 EC50 > 25000 nM T86591 C0VLP9 44564900 EC50 > 15000 nM T86591 C3K9RE 44564901 IC50 = 7290 nM T86591 CBF4N6 44564946 EC50 > 15000 nM T86591 CE16SW 44564947 EC50 = 4020 nM T86591 CEOU52 44565005 IC50 = 280 nM T86591 C9KRL0 44565006 IC50 = 3350 nM T86591 CIY78Z 44565059 EC50 = 11 nM T86591 C90ZGD 44571467 EC50 = 44 nM T86591 CC5D2Q 44571468 EC50 = 34 nM T86591 CJ1U6C 44571517 EC50 = 0.0038 nM T86591 CS1M8O 44571518 EC50 = 2 nM T86591 CO5I8F 44571519 EC50 = 1 nM T86591 C9MRZ4 44577533 EC50 = 1.09 nM T86591 CK32HI 44577534 EC50 = 0.272 nM T86591 C7QHB2 44577535 EC50 = 0.089 nM T86591 CGF48S 44577684 EC50 = 0.6 nM T86591 C72EIS 44577685 EC50 = 0.03 nM T86591 CBX3M7 44577687 EC50 = 4.2 nM T86591 CSZ15V 44579211 EC50 = 5980 nM T86591 C6NPQ1 44579212 EC50 = 3240 nM T86591 CA9V0O 44579252 EC50 = 7720 nM T86591 CJM4Q7 44579253 EC50 = 3400 nM T86591 CW91PX 44579254 EC50 = 3120 nM T86591 C1E0AL 44579255 EC50 = 542 nM T86591 CWT1Z0 44579288 EC50 = 2230 nM T86591 CJ82SN 44579289 EC50 = 11300 nM T86591 CV2W1S 44579290 EC50 = 17300 nM T86591 C8NIJ4 44579291 EC50 = 18100 nM T86591 C0GH1U 44579338 EC50 = 7580 nM T86591 C6S4IV 44579339 EC50 = 2080 nM T86591 C1Y4EU 44579340 EC50 = 64 nM T86591 C3JM1U 44579341 EC50 = 1120 nM T86591 C4ZX3L 44579390 EC50 = 1120 nM T86591 C45FJV 44579391 EC50 = 1150 nM T86591 CE1LR6 44579392 EC50 = 615 nM T86591 CS8N1U 44579393 EC50 = 2990 nM T86591 CU7FR4 44579432 EC50 = 10200 nM T86591 C5A2XS 44579433 EC50 = 8580 nM T86591 C1DJ9V 44579434 EC50 = 3670 nM T86591 C9P4VB 44579435 EC50 = 7670 nM T86591 CLF57W 44579436 EC50 = 9800 nM T86591 C0H9TA 44579477 EC50 = 9790 nM T86591 C0KI2H 44579478 EC50 = 1700 nM T86591 C10IXM 44579479 EC50 = 3860 nM T86591 C75KTS 44579480 EC50 = 25480 nM T86591 C6R9MQ 44579552 EC50 = 868 nM T86591 C7LE5D 44579553 EC50 = 331 nM T86591 CO5RI6 44587736 EC50 = 13 nM T86591 C15RIM 44587737 EC50 = 7.1 nM T86591 CVI68J 44587738 EC50 = 17 nM T86591 CO3IQ1 44587769 EC50 = 7.5 nM T86591 CNI3D6 44587770 EC50 = 13 nM T86591 CW67EM 44587801 EC50 = 200 nM T86591 C5JNC0 44589628 EC50 = 15000 nM T86591 CTWU08 44589804 EC50 = 2120 nM T86591 C5ND1E 44589805 EC50 = 1650 nM T86591 C92WZN 44589847 EC50 = 4490 nM T86591 CH5E9L 44589848 EC50 = 2180 nM T86591 CYQ8C5 44589849 EC50 = 2250 nM T86591 CD7ZA0 44589850 EC50 = 9250 nM T86591 CK8L4M 44589851 EC50 = 1430 nM T86591 CUL14S 44589898 EC50 = 2490 nM T86591 C2BW0J 44589899 EC50 = 1140 nM T86591 C1UQG8 44589954 EC50 = 2230 nM T86591 C35GSR 44589955 EC50 = 1100 nM T86591 CK0A4I 44589956 EC50 = 2810 nM T86591 CAMT56 44589957 EC50 = 350 nM T86591 C76GCX 44589958 EC50 = 450 nM T86591 CK34ZS 44590001 EC50 = 700 nM T86591 CH0WD8 44590002 EC50 = 27 nM T86591 C2I9QA 44590003 EC50 = 49 nM T86591 C4UM8I 44590004 EC50 = 65 nM T86591 C8WSC0 44590101 EC50 = 420 nM T86591 C5JW0E 44591474 EC50 = 284 nM T86591 CAZD19 44591655 IC50 = 294 nM T86591 CV3EF4 44591696 EC50 = 123 nM T86591 CI2PD6 44591724 EC50 = 2 nM T86591 COY5U4 44591725 EC50 = 43 nM T86591 CJ6H8E 44591726 EC50 = 20 nM T86591 C68RUE 44591751 EC50 = 27 nM T86591 C08IUA 44591752 EC50 = 13 nM T86591 CBUF12 44591753 EC50 = 555 nM T86591 CJY09Q 44591777 EC50 = 89 nM T86591 C3B5QX 44591778 EC50 = 27 nM T86591 CQH38Y 44591779 EC50 = 167 nM T86591 CQI2P9 44591780 EC50 = 16 nM T86591 CU49SN 44591801 EC50 = 1910 nM T86591 CY59XQ 44591802 EC50 = 358 nM T86591 C0S2NU 44591803 EC50 = 11 nM T86591 CTDI10 44591804 EC50 = 11 nM T86591 CYEN80 44591805 IC50 = 429 nM T86591 C3F5GK 44591814 EC50 = 650 nM T86591 CN3WH7 44591815 IC50 = 28 nM T86591 C7RNC3 44591816 EC50 = 58 nM T86591 CL6FI5 44591830 EC50 > 10000 nM T86591 CH9CK4 44626477 EC50 > 10000 nM T86591 CPW57V 44626478 EC50 > 10000 nM T86591 CUY95T 44626479 EC50 > 10000 nM T86591 CI31DJ 44626480 EC50 > 10000 nM T86591 C8TD4Z 44626481 EC50 > 10000 nM T86591 C0Z3XM 44626583 EC50 > 10000 nM T86591 C3VF6I 44626585 EC50 > 10000 nM T86591 C3ME5P 44626586 EC50 > 10000 nM T86591 CDIP96 44626587 EC50 > 10000 nM T86591 C6V4SD 44626689 EC50 > 10000 nM T86591 CB0GJ9 44626691 EC50 > 10000 nM T86591 CP9YH7 44626696 EC50 > 10000 nM T86591 C01AMG 44626697 EC50 > 10000 nM T86591 CY3I4V 44626789 EC50 > 10000 nM T86591 CXI58P 44626791 EC50 > 10000 nM T86591 C4JRP9 44626797 EC50 > 10000 nM T86591 C3YK1M 44626798 EC50 > 10000 nM T86591 C3Q2XF 44626799 EC50 > 10000 nM T86591 CB1ZX0 44626800 EC50 > 10000 nM T86591 C4A0WS 44626801 EC50 > 10000 nM T86591 C6EF1Q 44626888 EC50 > 10000 nM T86591 C6X8KS 44626889 EC50 > 10000 nM T86591 C5I8NM 44626890 EC50 > 10000 nM T86591 C8V9SP 44626891 EC50 > 10000 nM T86591 CTY31Z 44626892 EC50 > 10000 nM T86591 CQI69K 44626986 EC50 > 10000 nM T86591 C8NAD5 44626987 EC50 > 10000 nM T86591 C0RAL3 44626988 EC50 > 10000 nM T86591 C4BNA9 44626989 EC50 = 5200 nM T86591 CQ5O3I 44626990 EC50 > 10000 nM T86591 CESB05 44627078 EC50 = 5350 nM T86591 CSW84C 44627079 EC50 = 5250 nM T86591 C3ZM7B 44627080 EC50 = 2370 nM T86591 C6B2RO 44627083 EC50 > 10000 nM T86591 C2JB5Y 44627084 EC50 > 10000 nM T86591 CABC27 44627085 EC50 > 10000 nM T86591 CPS63M 44627086 EC50 = 690 nM T86591 CX41JP 44627087 EC50 = 1590 nM T86591 CL34OS 44627188 EC50 = 2600 nM T86591 CCQ59P 44627190 EC50 = 910 nM T86591 CMG9Q4 44627191 EC50 > 10000 nM T86591 C9OI6W 44627192 EC50 > 10000 nM T86591 CQJ26Z 44627297 EC50 > 10000 nM T86591 C87MHR 44627298 EC50 = 4080 nM T86591 C5W3IT 44627299 EC50 > 10000 nM T86591 CS25FR 44627300 EC50 > 10000 nM T86591 C0SYJ8 44627301 EC50 > 10000 nM T86591 CY49NK 44627302 EC50 > 10000 nM T86591 C6RBQ1 44627303 EC50 > 10000 nM T86591 CUL63M 44627304 EC50 > 10000 nM T86591 C1G2QK 44627305 EC50 > 10000 nM T86591 C96QCO 44627306 EC50 = 1990 nM T86591 CR8A1I 44627407 EC50 > 10000 nM T86591 CE2J5V 44627408 EC50 = 480 nM T86591 C43ZOX 44627409 EC50 > 10000 nM T86591 C7K0GI 44627410 EC50 > 10000 nM T86591 CA31WU 44627411 EC50 > 10000 nM T86591 CPY46S 44627412 EC50 > 10000 nM T86591 CI1VN2 44627413 EC50 > 10000 nM T86591 CK83HR 44627414 EC50 > 10000 nM T86591 C1DQ7N 44627415 EC50 > 10000 nM T86591 CF1Q5E 44627416 EC50 > 10000 nM T86591 CPFN63 44627417 EC50 = 1200 nM T86591 C9TNL0 44627524 EC50 > 10000 nM T86591 C3OXU2 44627525 EC50 > 10000 nM T86591 C3PZ6T 44627526 EC50 > 10000 nM T86591 CD47HB 44627527 EC50 > 10000 nM T86591 C1KAJ2 44627528 EC50 > 10000 nM T86591 CR93CX 44627529 EC50 = 410 nM T86591 CY95DP 44627531 EC50 > 10000 nM T86591 CD8L4U 44627532 EC50 > 10000 nM T86591 CYJ52X 44627533 EC50 > 10000 nM T86591 CJ43OZ 44627627 EC50 > 10000 nM T86591 CEA3I2 44627628 EC50 > 10000 nM T86591 CW7PG6 44627633 EC50 > 10000 nM T86591 CX0Q2Y 44627634 EC50 = 1090 nM T86591 CIWZ13 44627635 EC50 > 10000 nM T86591 CA4W0L 44627636 EC50 > 10000 nM T86591 C28SEU 44627637 EC50 > 10000 nM T86591 C6D0XF 44627728 EC50 > 10000 nM T86591 CAQ41R 44627729 EC50 > 10000 nM T86591 CCN8S2 44627730 EC50 > 10000 nM T86591 CGO41A 44627731 EC50 > 10000 nM T86591 C1HMU7 44627732 EC50 > 10000 nM T86591 C8K3GF 44627733 EC50 > 10000 nM T86591 C3T1HB 44627734 EC50 > 10000 nM T86591 CE93BG 44627735 EC50 > 10000 nM T86591 CPFV72 44627838 EC50 > 10000 nM T86591 CEH41N 44627839 EC50 > 10000 nM T86591 C2SJ5A 44627840 EC50 > 10000 nM T86591 C53AJB 44627841 EC50 > 10000 nM T86591 CXHP05 44627842 EC50 > 10000 nM T86591 CZL75R 44627843 EC50 > 10000 nM T86591 CRI4Q6 44627844 EC50 > 10000 nM T86591 CK7Z9X 44627845 EC50 > 10000 nM T86591 C95MPI 44627846 EC50 > 10000 nM T86591 C8SPR5 44627847 EC50 > 10000 nM T86591 C2LI9T 44627941 EC50 > 10000 nM T86591 CA8CB6 44627942 EC50 > 10000 nM T86591 CSDF01 44627943 EC50 > 10000 nM T86591 CM5D8L 44627944 EC50 > 10000 nM T86591 CX23ZO 44627945 EC50 > 10000 nM T86591 C35WJV 44627946 EC50 > 10000 nM T86591 CP9G7C 44627948 EC50 = 700 nM T86591 C6JXF9 44628046 EC50 > 10000 nM T86591 CQX2E8 44628047 EC50 > 10000 nM T86591 CW2I4H 44628048 EC50 > 10000 nM T86591 CUHD90 44628049 EC50 > 10000 nM T86591 C24MHW 44628050 EC50 > 10000 nM T86591 CI7SM1 45104339 IC50 > 10000 nM T86591 C0OX9J 45104340 IC50 > 10000 nM T86591 CB7ED5 45104341 IC50 > 10000 nM T86591 CLFU74 45104342 IC50 > 10000 nM T86591 COD76Z 45104343 IC50 > 10000 nM T86591 CGB9R5 45104439 IC50 > 10000 nM T86591 CNEV35 45104440 IC50 > 10000 nM T86591 CP7L6H 45104441 IC50 > 10000 nM T86591 CF1Y2V 45104442 IC50 > 10000 nM T86591 C8L5CG 45104443 IC50 > 10000 nM T86591 CRIS28 45104444 IC50 > 10000 nM T86591 CTWC94 45104445 IC50 > 10000 nM T86591 C4KRT0 45254002 EC50 = 8 nM T86591 CVL46G 45263732 EC50 = 35 nM T86591 CSLZ04 45267718 EC50 = 90 nM T86591 C0R8MQ 45267726 EC50 = 2000 nM T86591 CK31XL 45268054 EC50 = 34 nM T86591 C4A7GC 45268062 EC50 = 1000 nM T86591 C8AXK3 45268597 EC50 = 25 nM T86591 C0F7RJ 45268611 EC50 = 1500 nM T86591 C1EIF5 45269442 EC50 = 550 nM T86591 CU91HN 45269452 EC50 = 110 nM T86591 C74OGR 45269453 EC50 = 13800 nM T86591 CS7EC0 45269787 EC50 = 9 nM T86591 C4X8NT 45270286 EC50 = 150 nM T86591 CJC3M7 45270291 EC50 = 220 nM T86591 CTX61C 45271105 EC50 = 1700 nM T86591 C5U8HX 45271112 EC50 = 390 nM T86591 CZU9Q3 45271445 EC50 = 10000 nM T86591 CR1QU8 45271974 EC50 = 290 nM T86591 CN4ET7 45271983 EC50 = 250 nM T86591 CH92UP 45271992 EC50 = 49 nM T86591 CNU0H3 45272171 EC50 > 3000 nM T86591 C42QTW 45272810 EC50 = 85 nM T86591 CVU12R 45272820 EC50 = 190 nM T86591 CXS0Y5 45273207 EC50 = 73 nM T86591 COP75F 45273770 EC50 = 56 nM T86591 CQ4GE9 45273780 EC50 = 600 nM T86591 CM3Q4K 45482771 EC50 = 107 nM T86591 CY81ZP 45488162 EC50 = 300 nM T86591 C72CNH 45783216 Ki = 9100 nM T86591 C89QTJ 46184983 EC50 > 50000 nM T86591 CFA6V5 46196683 EC50 = 7.5 nM T86591 C9JV0C 46196684 EC50 = 9.2 nM T86591 CB4MV0 46196685 EC50 = 12.5 nM T86591 CJG9N2 46196686 EC50 = 6.3 nM T86591 C9ZV8D 46196687 EC50 = 6 nM T86591 C1GER0 46197994 EC50 = 289.3 nM T86591 CMJ12Z 46197995 EC50 = 39.1 nM T86591 CEGI58 46197996 EC50 = 16.5 nM T86591 CYAI40 46198106 EC50 = 122 nM T86591 CTI0F8 46198107 EC50 = 101 nM T86591 CJ9OY8 46198108 EC50 = 90 nM T86591 CI9QH8 46198109 EC50 = 68 nM T86591 CU3VQ1 46198110 EC50 = 134 nM T86591 C2P9ST 46198216 EC50 = 20.5 nM T86591 C3NFH5 46198217 EC50 = 10 nM T86591 CWR39G 46198218 EC50 = 340 nM T86591 CV8B3T 46198219 EC50 = 108 nM T86591 CSEL57 46198325 EC50 = 37 nM T86591 C2VIF3 46198326 EC50 = 15.8 nM T86591 C6JWH5 46198327 EC50 = 9.1 nM T86591 CIJN79 46198328 EC50 = 8.7 nM T86591 C13RUW 46198329 EC50 = 12 nM T86591 CY97NP 46213107 EC50 > 10000 nM T86591 C5D9KI 46216831 EC50 = 10 nM T86591 CS4K6Y 46216832 EC50 = 5 nM T86591 CF80GU 46228280 EC50 > 100000 nM T86591 C5E2FZ 46228281 EC50 > 100000 nM T86591 CJ6AN0 46229742 EC50 = 2300 nM T86591 C0ZWT3 46229787 EC50 = 50 nM T86591 C2VBA4 46229788 EC50 = 50 nM T86591 CT9JR4 46229789 EC50 = 400 nM T86591 COI07L 46229832 EC50 = 2400 nM T86591 C7M2LT 46229833 EC50 = 500 nM T86591 C2C4EF 46229834 EC50 = 20 nM T86591 C2OCX1 46229835 EC50 = 30 nM T86591 C3DY0A 46229869 EC50 = 3 nM T86591 CFTW35 46229870 EC50 = 100 nM T86591 CNE12J 46229871 EC50 = 2 nM T86591 C1O2HJ 46229903 EC50 = 400 nM T86591 C2R8WH 46232959 EC50 > 10000 nM T86591 C12JOZ 46232960 EC50 > 10000 nM T86591 CL36PQ 46233001 EC50 = 4960 nM T86591 C3Q6DN 46233002 EC50 > 10000 nM T86591 C0P5ED 46233003 EC50 > 10000 nM T86591 C19XSC 46233038 EC50 > 10000 nM T86591 CBSA69 46233039 EC50 > 10000 nM T86591 C5O7FJ 46233040 EC50 = 6140 nM T86591 CE93XQ 46233070 EC50 > 10000 nM T86591 C9A2QS 46233071 EC50 > 10000 nM T86591 CT53DY 46233072 EC50 > 10000 nM T86591 CVZ97H 46861800 EC50 = 13 nM T86591 CE72MC 46878644 EC50 > 10000 nM T86591 C4WDX1 46878645 EC50 = 300 nM T86591 C1QT8Z 46878727 EC50 = 800 nM T86591 CWZ8N4 46878728 EC50 = 840 nM T86591 C4WO1G 46878729 EC50 = 1060 nM T86591 CRK26D 46878777 EC50 > 10000 nM T86591 C0HYG2 46878778 EC50 > 10000 nM T86591 C49SRK 46878779 EC50 > 10000 nM T86591 C62JTF 46878780 EC50 > 10000 nM T86591 C3OZP9 46878781 EC50 = 1150 nM T86591 C51RAC 46878843 EC50 > 10000 nM T86591 CQ7JI0 46879867 EC50 = 790 nM T86591 CDL01S 46880009 IC50 = 10 nM T86591 C8I4CV 46880010 EC50 = 3000 nM T86591 C9T0FX 46880011 EC50 = 130 nM T86591 CFMH58 46880012 EC50 = 120 nM T86591 CQF9J7 46880049 EC50 = 570 nM T86591 CG3D5X 46880447 EC50 > 10000 nM T86591 CD05FS 46884868 EC50 > 100000 nM T86591 CF65OR 46888895 EC50 = 64 nM T86591 C0S8WL 46888896 EC50 = 68 nM T86591 CB3FC1 46888897 EC50 = 29.9 nM T86591 C5MH4J 46888966 EC50 = 235 nM T86591 CIQT59 46888967 EC50 = 1225 nM T86591 CRJ67A 46888968 EC50 = 451 nM T86591 C20VWR 46888969 EC50 = 1086 nM T86591 CGI9Q8 46888992 EC50 = 395 nM T86591 C3ZG7B 46888993 EC50 = 73 nM T86591 C2MO0J 46888994 EC50 = 87 nM T86591 CJB37Y 46888995 EC50 = 90 nM T86591 C4N7ZM 46889020 EC50 = 41.8 nM T86591 CV0O3M 46889021 EC50 = 304 nM T86591 C0IVK1 46889022 EC50 = 1453 nM T86591 CCNZ52 46889045 EC50 > 2500 nM T86591 CZ1H2N 46889046 EC50 = 145 nM T86591 CU9R0D 46889047 EC50 = 22 nM T86591 C6TQX2 46889072 EC50 = 66 nM T86591 CJ3V7K 46889073 EC50 = 471 nM T86591 CQJ70A 46889074 EC50 = 51 nM T86591 CVPM17 46890332 EC50 = 1000 nM T86591 CIU0K4 46890333 EC50 = 700 nM T86591 CKB7C4 46890417 EC50 = 900 nM T86591 C0KAC2 46890418 EC50 = 1000 nM T86591 CEHW01 46890419 EC50 = 10000 nM T86591 CGC6X0 46890420 EC50 > 25000 nM T86591 CGF2M3 46890461 EC50 = 2000 nM T86591 CTF76Z 46890462 EC50 = 300 nM T86591 CS12HI 46890463 EC50 = 3000 nM T86591 C6JR1Z 46890509 EC50 = 1500 nM T86591 CF7TS3 46890510 EC50 > 25000 nM T86591 CO6ED2 46890511 EC50 = 13000 nM T86591 CHCO92 46890512 EC50 = 7000 nM T86591 C0H6FU 46908722 EC50 > 10000 nM T86591 CL0R6B 46908814 EC50 > 10000 nM T86591 C4FAD6 46908815 EC50 > 10000 nM T86591 CI7U3G 46908816 EC50 > 10000 nM T86591 C2QIR9 46908817 EC50 > 10000 nM T86591 CRF0E4 46908818 EC50 > 10000 nM T86591 C6VB0S 46908904 EC50 > 10000 nM T86591 C3NMP1 46908905 EC50 > 10000 nM T86591 CN9L7G 46916268 EC50 > 15000 nM T86591 CS13YQ 49846481 IC50 > 100000 nM T86591 CUD91T 49862248 EC50 = 680000 nM T86591 CZ9UD6 50901657 IC50 > 250000 nM T86591 CP3Y0J 50925503 EC50 = 350.3 nM T86591 CD2G5X 50925504 EC50 = 24.6 nM T86591 C4PK6S 50942697 EC50 = 2500 nM T86591 C96HOP 50942698 EC50 = 1250 nM T86591 CK03LY 51038993 EC50 = 13800 nM T86591 CT59YM 51039006 EC50 = 8600 nM T86591 CNVB53 51346913 EC50 = 120 nM T86591 CAXJ10 52918120 IC50 = 10000 nM T86591 CRN19G 52918121 IC50 = 7943.28 nM T86591 C3VEH4 52941520 EC50 = 4000 nM T86591 C4KQR2 52948223 EC50 = 4200 nM T86591 C3KM6T 53233135 EC50 = 0.00031 nM T86591 CN8H7B 53240432 EC50 = 2400 nM T86591 CL83BY 53317593 EC50 > 1000 nM T86591 CVN51I 53317892 EC50 = 15.2 nM T86591 CTUA27 53317893 EC50 = 83.1 nM T86591 C4H5CJ 53319204 EC50 = 21000 nM T86591 C7I9UO 53319246 EC50 = 39.4 nM T86591 C1JIB3 53319416 EC50 > 30000 nM T86591 C8JL7M 53323370 EC50 = 6300 nM T86591 C3PYV7 53325836 EC50 = 120 nM T86591 CSQM04 53356799 EC50 = 743 nM T86591 C3PL6K 53380705 EC50 = 50600 nM T86591 CA5BC0 53380706 IC50 = 6500 nM T86591 CT9QZ3 53380805 IC50 = 22200 nM T86591 C39CYS 53380806 IC50 = 19900 nM T86591 CL2VM8 54579977 IC50 = 10000 nM T86591 CV9U5K 54580014 IC50 = 12589.25 nM T86591 C9IN5X 54580015 IC50 = 19952.62 nM T86591 C64SWC 54580016 IC50 = 19952.62 nM T86591 C76WZO 54580529 EC50 = 60 nM T86591 C6M9HP 54580530 EC50 = 15 nM T86591 CKBG47 54580531 EC50 = 29 nM T86591 CSH41U 54580814 EC50 = 2300 nM T86591 C8MLC0 54580964 IC50 = 6309.57 nM T86591 C8EUF2 54580965 IC50 = 10000 nM T86591 CM6I8P 54580966 IC50 = 15848.93 nM T86591 CR5DC6 54580967 IC50 = 19952.62 nM T86591 CPT96V 54581011 IC50 = 7943.28 nM T86591 C2E5NY 54581038 EC50 > 10000 nM T86591 CM95BU 54581270 IC50 = 46.99 nM T86591 C81THX 54581535 EC50 = 5 nM T86591 CBE79V 54581857 EC50 = 34100 nM T86591 CAT03Y 54582018 IC50 = 19952.62 nM T86591 CMLX87 54582047 IC50 = 10000 nM T86591 CRKL15 54582795 EC50 = 13900 nM T86591 CT4IJ9 54582796 EC50 = 830 nM T86591 CQ89ZY 54582993 IC50 = 19952.62 nM T86591 CP92OU 54582994 IC50 = 12589.25 nM T86591 CGTN92 54582995 IC50 = 12589.25 nM T86591 CHQ79P 54583754 EC50 = 14700 nM T86591 C1D5YV 54583795 EC50 = 13200 nM T86591 CK48SJ 54583995 IC50 = 10000 nM T86591 C9YDX0 54583996 IC50 = 15848.93 nM T86591 CX1V3U 54583997 IC50 = 12589.25 nM T86591 CGXM65 54583998 IC50 = 10000 nM T86591 CK6CI7 54584935 IC50 = 12589.25 nM T86591 C1KOF7 54584936 IC50 > 25118.86 nM T86591 CPXG09 54584937 IC50 = 19952.62 nM T86591 CBO34V 54584938 IC50 = 10000 nM T86591 C02CRJ 54584979 EC50 > 10000 nM T86591 CNO4C1 54585198 IC50 = 19 nM T86591 CQU27M 54585710 EC50 > 10000 nM T86591 C4DX7E 54585711 EC50 = 3300 nM T86591 C3TU7R 54585867 IC50 = 15848.93 nM T86591 COX28A 54585896 IC50 = 15848.93 nM T86591 C6ZSM0 54585897 IC50 = 15848.93 nM T86591 CXL71T 54585898 IC50 = 10000 nM T86591 C7D1LE 54585899 IC50 = 15848.93 nM T86591 C0I2DH 54585900 IC50 > 19952.62 nM T86591 CP8F9I 54585901 IC50 = 12589.25 nM T86591 C0JOG1 54585902 IC50 = 19952.62 nM T86591 C9Q0VG 54585903 IC50 = 15848.93 nM T86591 CU43ME 54585904 IC50 = 15848.93 nM T86591 CFZ6E9 54585935 EC50 = 620 nM T86591 CO0XN5 54585936 EC50 = 3600 nM T86591 CW0L9M 54586395 EC50 = 3600 nM T86591 C6EC0W 54586396 EC50 = 52 nM T86591 CO0X2A 54586658 EC50 = 12900 nM T86591 CM9GL4 54586691 EC50 > 10000 nM T86591 C8NZ6D 54586832 IC50 = 15848.93 nM T86591 C18JYB 54586833 IC50 = 15848.93 nM T86591 C2K6FY 54586870 IC50 = 12589.25 nM T86591 C8UO7K 54586871 IC50 = 19952.62 nM T86591 CTL0F5 54586872 IC50 = 15848.93 nM T86591 C28UYH 54586873 IC50 = 10000 nM T86591 CF3BK8 54586906 EC50 = 3600 nM T86591 CP6D9X 54586907 EC50 = 3600 nM T86591 C7N0YU 54587410 EC50 = 41 nM T86591 C14QDZ 54587728 EC50 > 10000 nM T86591 C5J0BW 54587729 EC50 = 2900 nM T86591 C5ZX4B 54597874 EC50 > 10000 nM T86591 CUJ76C 54753638 EC50 = 11300 nM T86591 CPLG91 54753639 EC50 = 9300 nM T86591 CMS2T9 54753640 EC50 = 1000 nM T86591 C2HRN4 54753641 EC50 = 6600 nM T86591 CRN5D3 54764927 EC50 = 560 nM T86591 CC92QD 56641248 EC50 = 109300 nM T86591 CM3S7X 56641249 EC50 = 27100 nM T86591 CLTJ50 56641379 EC50 = 61500 nM T86591 C9X7QB 56641380 EC50 = 9100 nM T86591 C89YMG 56641381 EC50 = 43700 nM T86591 CKD6P8 56641774 EC50 = 18800 nM T86591 CKIC64 56659331 EC50 = 3400 nM T86591 CRB95Z 56659332 EC50 = 1800 nM T86591 C92XSL 56659333 EC50 = 1100 nM T86591 CT1A3Y 56659334 EC50 = 1700 nM T86591 CA9U3S 56659347 EC50 = 0.026 nM T86591 CF29WQ 56659348 EC50 = 0.00005 nM T86591 C4CP6U 56666265 EC50 = 6600 nM T86591 CIUN54 56666266 EC50 = 8900 nM T86591 C7NA3W 56666267 EC50 = 1700 nM T86591 CPQB39 56669679 EC50 = 33000 nM T86591 CGP42W 56669681 EC50 = 1400 nM T86591 C5I0GB 56669682 EC50 = 1700 nM T86591 C1MAL6 56669688 EC50 = 3 nM T86591 CVQ64B 56669689 EC50 = 0.1 nM T86591 C50PUC 56669690 EC50 = 0.00007 nM T86591 CN8YH0 56673196 EC50 = 22 nM T86591 C51FPO 56673531 IC50 = 27900 nM T86591 CH0KR3 56676514 EC50 = 29000 nM T86591 CQ58IX 56676515 EC50 = 14000 nM T86591 CV6Z3S 56676516 EC50 = 4500 nM T86591 C1H5IV 56676523 EC50 = 20 nM T86591 CX6B7G 56676845 IC50 = 31000 nM T86591 CN26ZO 56679837 EC50 = 11000 nM T86591 CA1O0N 56679838 EC50 = 2500 nM T86591 CV12UQ 56679849 EC50 = 0.00006 nM T86591 CKLC32 56679850 EC50 = 1.9 nM T86591 CXMR78 56925781 IC50 > 50000 nM T86591 C5HQZ6 56925892 IC50 > 50000 nM T86591 C0NRU5 56925893 IC50 > 50000 nM T86591 C2B6MF 56925894 IC50 > 50000 nM T86591 CJ46YQ 56925895 IC50 > 50000 nM T86591 CR6TP4 56925896 IC50 > 50000 nM T86591 CVO3A2 56925994 IC50 > 50000 nM T86591 CLCM62 56925995 IC50 > 50000 nM T86591 C8GLC1 56925996 IC50 > 50000 nM T86591 C2M8DR 56925997 IC50 > 50000 nM T86591 CD75ZU 56925998 IC50 > 50000 nM T86591 C8YGX7 56926094 IC50 > 50000 nM T86591 C15OKZ 56926095 IC50 > 50000 nM T86591 CN68DG 56926096 IC50 > 50000 nM T86591 C4K1XH 56926097 IC50 > 50000 nM T86591 CFO3R4 56926098 IC50 > 50000 nM T86591 C7X3WK 56926185 IC50 > 50000 nM T86591 CZEF98 56926186 IC50 > 50000 nM T86591 C92DPX 56926187 IC50 > 50000 nM T86591 CSJW15 56926188 IC50 > 50000 nM T86591 C9VTF3 56926189 IC50 > 50000 nM T86591 CMK92V 56926276 IC50 > 50000 nM T86591 COT54N 56929220 EC50 = 770 nM T86591 COP96Y 56929315 EC50 = 1760 nM T86591 CNB56J 56940812 EC50 > 10000 nM T86591 CA7Y1Z 56941393 EC50 > 10000 nM T86591 C1DQ4M 56942395 EC50 > 10000 nM T86591 CN5Z9T 56945389 EC50 = 25 nM T86591 CNC6B5 56945390 EC50 = 122 nM T86591 CI6L5H 56945391 EC50 = 1720 nM T86591 CRJC63 56945487 EC50 = 620 nM T86591 C0MC8V 56949691 EC50 > 10000 nM T86591 CQ19IH 56949692 EC50 > 10000 nM T86591 CB4F9K 56949693 EC50 > 10000 nM T86591 CWQY91 57345616 EC50 = 1000 nM T86591 CP89DR 57390390 EC50 = 4500 nM T86591 CCK42T 57390448 EC50 = 24800 nM T86591 C6SJH9 57390449 EC50 = 6500 nM T86591 CWMF02 57390810 EC50 = 1500 nM T86591 C9V4NS 57390811 EC50 > 3400 nM T86591 C9SB5K 57390812 EC50 = 72 nM T86591 C25WYC 57391048 EC50 > 3500 nM T86591 CIFN56 57391546 EC50 > 10000 nM T86591 C8Y0ET 57391547 EC50 > 10000 nM T86591 C96EIM 57392586 EC50 = 280 nM T86591 CT3U5R 57392587 EC50 = 120 nM T86591 CIVL69 57392628 EC50 = 1500 nM T86591 CX8QN1 57392629 EC50 = 53 nM T86591 C7A2XY 57392630 EC50 = 21 nM T86591 C5JD9O 57392836 EC50 = 700 nM T86591 C1FS9Q 57392837 EC50 = 4400 nM T86591 C5I1CA 57393296 EC50 > 10000 nM T86591 C5A7HW 57393297 EC50 > 10000 nM T86591 CB01SO 57393940 EC50 = 19000 nM T86591 C5BG1A 57394147 EC50 = 710 nM T86591 CK5HD6 57394349 EC50 = 850 nM T86591 CZ0Y1N 57394350 EC50 = 810 nM T86591 CX34SN 57394351 EC50 = 37 nM T86591 CHN65K 57394378 EC50 > 14000 nM T86591 C7Q3IB 57395028 EC50 > 10000 nM T86591 CT45EM 57395675 EC50 = 6600 nM T86591 CHM9Q5 57395750 EC50 = 22300 nM T86591 CHRX78 57396101 EC50 = 6 nM T86591 C9V1KC 57396779 EC50 > 10000 nM T86591 CQ71JU 57396780 EC50 > 10000 nM T86591 CLI70F 57396782 EC50 > 10000 nM T86591 C7YC4Z 57396783 EC50 > 10000 nM T86591 C1D7YR 57397473 EC50 = 10300 nM T86591 C5ZCT7 57397527 EC50 = 21000 nM T86591 C2DOZ9 57397718 EC50 = 735 nM T86591 C7JRE9 57397870 EC50 = 3400 nM T86591 C3O8JG 57398546 EC50 > 10000 nM T86591 C6ET7R 57398547 EC50 > 10000 nM T86591 C1DPW9 57398548 EC50 > 10000 nM T86591 C19KAD 57398549 EC50 > 10000 nM T86591 CKL3A8 57398721 EC50 = 100 nM T86591 C8HB5R 57399155 EC50 = 2500 nM T86591 CKYR74 57399206 EC50 = 9800 nM T86591 CPX5Z8 57399207 EC50 = 2200 nM T86591 CU6LA3 57399208 EC50 = 1400 nM T86591 C09OZX 57399558 EC50 = 700 nM T86591 CPV28C 57399559 EC50 = 810 nM T86591 CVO68Y 57399560 EC50 > 6000 nM T86591 C1T4AN 57399600 EC50 > 12000 nM T86591 CQT4G5 57400212 EC50 > 10000 nM T86591 CQC7F9 57400214 EC50 > 10000 nM T86591 CH5AK1 57400966 EC50 = 5100 nM T86591 CVXB34 57400967 EC50 = 5400 nM T86591 CXO3V1 57401284 EC50 = 2400 nM T86591 C82NSD 57401312 EC50 = 23 nM T86591 CTWX97 57402017 EC50 > 10000 nM T86591 C69PVW 57403073 EC50 = 26 nM T86591 CXA36C 57404419 EC50 > 60000 nM T86591 CS4J1B 57404439 EC50 = 19500 nM T86591 C1Y7WA 58754075 IC50 = 8912.51 nM T86591 CLOJ94 58977440 EC50 = 150 nM T86591 CT39UP 58977442 IC50 > 10000 nM T86591 CE0Y7W 58977463 EC50 = 1470 nM T86591 CN6G8S 58977476 EC50 = 1650 nM T86591 CDX3L4 58977524 EC50 = 850 nM T86591 C3L2SG 58977541 EC50 = 14 nM T86591 CW79RE 58977572 EC50 = 6 nM T86591 CWL7J2 58977618 IC50 > 10000 nM T86591 C0A6OI 58977630 EC50 = 2910 nM T86591 C1MDW5 58977670 IC50 > 10000 nM T86591 CMTB34 58977737 EC50 = 4410 nM T86591 CIAZ23 58977763 EC50 = 2580 nM T86591 CFUB93 58977773 EC50 = 2480 nM T86591 CSO5C6 58977817 IC50 = 660 nM T86591 CCS43U 58977846 EC50 = 20 nM T86591 CK6Y1Q 58977874 IC50 = 320 nM T86591 CI86BL 58977881 EC50 = 2590 nM T86591 C85QWJ 58977899 EC50 = 2870 nM T86591 C0X2IS 58977913 EC50 = 1000 nM T86591 CG1YR0 58977919 EC50 > 10000 nM T86591 CJQ4R7 59026512 EC50 > 15000 nM T86591 CP9E4V 59096898 EC50 = 1288.25 nM T86591 C79PXW 60166133 EC50 > 10000 nM T86591 COCI72 60166134 EC50 > 10000 nM T86591 CO2X7F 60166264 EC50 > 10000 nM T86591 CY31AP 60166265 EC50 > 10000 nM T86591 C38XJT 60166266 EC50 > 10000 nM T86591 CFA9N8 60166267 EC50 > 10000 nM T86591 CES4D2 60166268 EC50 > 10000 nM T86591 C3P5MV 60166383 EC50 > 10000 nM T86591 CR01ID 60166384 EC50 > 10000 nM T86591 C6U3KL 60166385 EC50 > 10000 nM T86591 CN78JU 60166386 EC50 > 10000 nM T86591 C7IW2B 60166387 EC50 > 10000 nM T86591 CC3HM4 60166513 EC50 > 10000 nM T86591 CL0V6S 60166514 EC50 > 10000 nM T86591 CON53Z 60166515 EC50 > 10000 nM T86591 CU2O0N 60166516 EC50 > 10000 nM T86591 CZ8VU0 60166647 EC50 > 10000 nM T86591 CYT71B 60166648 EC50 > 10000 nM T86591 CG71ZE 60166649 EC50 = 135.5 nM T86591 CC4YD6 60166650 EC50 = 35 nM T86591 C3LGI6 60166651 EC50 = 591.7 nM T86591 CALX08 60166891 EC50 = 861.3 nM T86591 CD6RH2 66560742 EC50 = 6000 nM T86591 C5FAY1 66561969 EC50 = 4000 nM T86591 C2RDZ8 68002585 EC50 = 34500 nM T86591 C9RO7Z 68588383 EC50 = 5.8 nM T86591 C2SVJ4 68661324 EC50 > 10000 nM T86591 C0XIR1 68661491 EC50 > 10000 nM T86591 CE25MB 68661514 EC50 > 10000 nM T86591 CAK3E0 68661534 EC50 > 10000 nM T86591 CZ64KE 68661565 EC50 > 10000 nM T86591 CGN64W 68661587 EC50 > 10000 nM T86591 CXT3L7 68661602 EC50 > 10000 nM T86591 C1T8YF 68661621 EC50 > 10000 nM T86591 CELF49 68661767 EC50 > 10000 nM T86591 C5WPA0 68661793 EC50 > 10000 nM T86591 CE9T6Z 68661809 EC50 > 10000 nM T86591 CC1W7Z 68661980 EC50 > 10000 nM T86591 CNJA68 68661986 EC50 > 10000 nM T86591 C6NEB4 68662059 EC50 > 10000 nM T86591 CF57AT 68662065 EC50 > 10000 nM T86591 C81RYD 68662112 EC50 > 10000 nM T86591 CS5K4W 68662136 EC50 > 10000 nM T86591 CV1LZ7 68662186 EC50 > 10000 nM T86591 CT18SJ 68662238 EC50 > 10000 nM T86591 C1WL3P 68674744 EC50 = 260 nM T86591 CKM6E9 68675602 EC50 = 160 nM T86591 CS4V7A 68676158 EC50 > 5000 nM T86591 C9PF1U 68676459 EC50 > 5000 nM T86591 CH62WK 68676471 EC50 = 305 nM T86591 CM1O9L 68676633 EC50 = 419 nM T86591 CE9IP3 68676761 EC50 = 901 nM T86591 CI7DX4 68676782 EC50 = 2360 nM T86591 CFN69J 68677403 EC50 = 956 nM T86591 CIYO07 68677705 EC50 > 5000 nM T86591 CIU96H 68677842 EC50 = 1537 nM T86591 C6HY5N 68809763 EC50 = 30600 nM T86591 CL27US 68811733 EC50 = 75100 nM T86591 CZ3WJ6 70680568 EC50 = 12 nM T86591 CUN9B1 70680569 EC50 = 100 nM T86591 CY9GZ8 70681800 IC50 = 1324.34 nM T86591 C2DZ3G 70681801 IC50 = 1845.02 nM T86591 CSEF42 70681805 IC50 = 60.95 nM T86591 CMT6J3 70681806 IC50 = 2642.41 nM T86591 C9TUJ1 70682504 EC50 = 60 nM T86591 C8LN6Z 70683449 EC50 = 1480 nM T86591 CB4A7U 70683915 IC50 = 473.15 nM T86591 CTD3I6 70685551 EC50 = 971 nM T86591 C7TJC3 70686048 IC50 = 1106 nM T86591 C13CJK 70686054 IC50 = 629.51 nM T86591 CCBM25 70688041 IC50 = 2080 nM T86591 CEL43F 70688075 EC50 = 432.4 nM T86591 C40KCB 70688165 IC50 = 219.79 nM T86591 CFY6Z4 70688166 IC50 = 339.63 nM T86591 CP72KL 70688172 IC50 = 352.37 nM T86591 CR52NL 70689089 IC50 = 0.28 nM T86591 CYJ75M 70690069 IC50 = 7470 nM T86591 CIC8V5 70690196 IC50 = 10889.3 nM T86591 C69MGD 70692364 IC50 = 125.03 nM T86591 C34KXB 70692371 IC50 = 41.98 nM T86591 CR2YQ9 70693621 EC50 = 46100 nM T86591 C4T9MB 70693933 EC50 = 887 nM T86591 C90MIS 70694287 IC50 = 2820 nM T86591 C5C9HR 70694419 IC50 = 95.06 nM T86591 C4DRC8 70694428 IC50 = 36.98 nM T86591 C29DRB 70694429 IC50 = 89.95 nM T86591 CCSX40 70695398 IC50 = 0.59 nM T86591 CV3T4P 70695727 EC50 > 60000 nM T86591 CR2PJ4 70695728 EC50 = 53200 nM T86591 CIZ7O3 70696377 EC50 = 14000 nM T86591 CL0JN8 70696489 IC50 = 809.1 nM T86591 C90GXS 70696490 IC50 = 39.99 nM T86591 C9X1JF 71449115 EC50 = 1100 nM T86591 C9PA6Y 71449654 EC50 > 50000 nM T86591 CL8W1E 71450437 EC50 = 36 nM T86591 CDVK19 71450438 EC50 = 13 nM T86591 CZO16C 71450439 EC50 > 25000 nM T86591 CK5WV7 71450440 EC50 = 500 nM T86591 CC5T1Z 71450448 EC50 = 600 nM T86591 C2TLF8 71450909 EC50 = 300 nM T86591 C2XRH5 71451339 IC50 = 600 nM T86591 C6MH9R 71451340 EC50 = 7100 nM T86591 CGN2A9 71452269 EC50 = 32 nM T86591 CQY90O 71452270 EC50 > 25000 nM T86591 CAR5V4 71452275 EC50 = 45800 nM T86591 CM63BE 71452661 EC50 = 70 nM T86591 CS45JB 71452719 EC50 = 9600 nM T86591 CSN6G2 71452725 EC50 = 1399 nM T86591 CGF2U1 71453153 IC50 = 480 nM T86591 C0I1QS 71453154 IC50 = 46500 nM T86591 C9ERN1 71453290 EC50 = 47100 nM T86591 CP27KN 71454069 EC50 = 26 nM T86591 CT27RV 71454077 EC50 = 40500 nM T86591 CY7UG1 71454437 EC50 = 1600 nM T86591 C5US2A 71455005 EC50 > 50000 nM T86591 CU34JE 71455800 EC50 = 8.1 nM T86591 CRQA20 71455801 EC50 = 56 nM T86591 CIZA80 71455811 EC50 = 64000 nM T86591 C8PBI3 71456242 EC50 = 100 nM T86591 C3RB2L 71456252 EC50 = 7.3 nM T86591 CMYN63 71456672 EC50 = 1590 nM T86591 CW07PO 71456673 IC50 = 900 nM T86591 CK9YX1 71457371 EC50 = 5000 nM T86591 CJ5WR8 71457584 EC50 = 9 nM T86591 C4O7MV 71457585 EC50 = 5.1 nM T86591 CU49YK 71457599 EC50 = 5600 nM T86591 CM4F2S 71457600 EC50 = 18300 nM T86591 C9GET3 71458051 EC50 = 1300 nM T86591 CRF20V 71458052 EC50 = 1086 nM T86591 C8LPE5 71458512 IC50 = 5100 nM T86591 CDI27W 71458513 EC50 = 10700 nM T86591 C26UVB 71458514 IC50 = 68500 nM T86591 C16BJE 71459228 EC50 = 7000 nM T86591 CC17GK 71459487 EC50 = 3.9 nM T86591 CWO9U1 71459496 EC50 = 9900 nM T86591 C4EB3N 71459497 EC50 = 42800 nM T86591 C9RB3Y 71459933 EC50 = 1200 nM T86591 C2LG7J 71459934 EC50 = 200 nM T86591 C9D0SN 71460357 IC50 = 600 nM T86591 C1FP8C 71461220 EC50 = 1.7 nM T86591 CQW65K 71461221 EC50 = 5200 nM T86591 C0ZM1O 71461231 EC50 = 11600 nM T86591 CX1SC6 71461648 EC50 = 1100 nM T86591 CGF67V 71462737 EC50 = 6000 nM T86591 C6O0TB 71462957 EC50 = 670 nM T86591 CAH63D 71462958 EC50 = 10000 nM T86591 CY6A5T 71462959 EC50 = 7200 nM T86591 CTCS46 71462964 EC50 = 44600 nM T86591 CO64EH 71544680 EC50 = 210 nM T86591 C0AV4J 71544681 EC50 = 220 nM T86591 C72FAV 71544682 EC50 = 67 nM T86591 CS56TM 71544683 EC50 = 31 nM T86591 CJ93XY 71544684 EC50 = 120 nM T86591 CKTE38 71544685 EC50 = 22 nM T86591 C9BXE3 71544686 EC50 = 44 nM T86591 CLS10T 71544851 EC50 = 130 nM T86591 C3GWQ1 71544852 EC50 = 12 nM T86591 C4UV5P 71544853 EC50 = 240 nM T86591 CVB90J 71544854 EC50 = 500 nM T86591 CR0C9E 71544855 EC50 = 280 nM T86591 CFZ3A6 71547107 EC50 = 990 nM T86591 CT0ZA3 71547108 EC50 = 80 nM T86591 COVC32 71547109 EC50 = 1130 nM T86591 C4W5PD 71547110 EC50 = 2100 nM T86591 C6FZ7C 71547111 EC50 = 230 nM T86591 CL4A2V 71604423 EC50 = 17 nM T86591 C10SPC 71616170 EC50 = 186 nM T86591 CNPK13 71616171 EC50 = 635 nM T86591 CI1LF2 71616173 EC50 = 64 nM T86591 C9U6VX 71616290 EC50 = 26 nM T86591 CK58CF 71616294 EC50 = 30 nM T86591 C6LT3W 71616409 EC50 = 652 nM T86591 C5NU0T 71721539 EC50 = 1400 nM T86591 CBN2H1 71735902 IC50 = 114 nM T86591 CA2IY6 71736703 IC50 = 113 nM T86591 CMFD46 72734874 EC50 = 6600 nM T86591 C2K0GM 72734875 EC50 = 6500 nM T86591 CBO3D4 72734876 EC50 = 3600 nM T86591 C3QIV9 72735053 EC50 = 8200 nM T86591 CWHB65 72735057 EC50 = 5700 nM T86591 CU07KO 72735238 EC50 = 2900 nM T86591 CX2ND4 72735418 EC50 = 3900 nM T86591 C4JSP6 72735591 EC50 = 5400 nM T86591 CFW41I 73167563 EC50 = 1050 nM T86591 CX20AE 73347299 EC50 = 588.84 nM T86591 CBSQ86 73347300 EC50 = 2511.89 nM T86591 C1GIP0 73347301 EC50 = 3019.95 nM T86591 CUZC61 73347302 EC50 = 3890.45 nM T86591 C0VHS6 73351898 EC50 = 2398.83 nM T86591 C93SWK 73351899 EC50 = 891.25 nM T86591 CUEA53 73356438 EC50 = 630.96 nM T86591 C57URV 76309038 EC50 = 1047 nM T86591 C8X4IT 76309039 EC50 = 6900 nM T86591 C49IUW 76311770 EC50 = 3.981 nM T86591 CJ4P7G 76312720 EC50 = 6456 nM T86591 C5X3HV 76312721 EC50 = 457 nM T86591 CGT93D 76319009 EC50 = 1 nM T86591 C75YZJ 76319010 EC50 = 2511.89 nM T86591 C32YPJ 76321033 EC50 = 21 nM T86591 CZ57LN 76326666 EC50 = 4168693.83 nM T86591 C23OFU 76330323 EC50 = 25003453.62 nM T86591 C78XLM 76330830 EC50 = 3467.37 nM T86591 CR6AG1 76334423 EC50 = 1288.25 nM T86591 CIW0C8 76334424 EC50 = 3600 nM T86591 CES0Z2 76335714 IC50 = 20800 nM T86591 C6X5MD 86279340 EC50 = 1960 nM T86591 C5WG3I 86582930 EC50 = 821 nM T86591 C63WUO 87537807 EC50 = 1263 nM T86591 C4YQ3K 89815987 IC50 = 218 nM T86591 CTBQ27 90469357 EC50 = 670 nM T86591 CR3I0E 90469358 EC50 > 100000 nM T86591 CY09NA 90469423 EC50 > 100000 nM T86591 C0GQ9R 90469424 EC50 > 100000 nM T86591 CSRZ25 90469425 EC50 = 6623 nM T86591 CZBS53 90469426 EC50 = 1978 nM T86591 CQK8E7 90656009 EC50 = 15700 nM T86591 C4BA8W 90656430 IC50 = 4800 nM T86591 CW7E1G 90656431 IC50 = 40 nM T86591 CR6E0Z 90656432 IC50 = 2.8 nM T86591 C5MI8N 90656433 IC50 = 13 nM T86591 CVDR97 90656434 IC50 = 34 nM T86591 CV1LC0 90656435 IC50 = 80 nM T86591 CYTD58 90656436 IC50 = 3 nM T86591 CML6N1 90656437 IC50 = 4.6 nM T86591 CF5S2W 90656438 IC50 = 6.6 nM T86591 CR0DZ3 90656439 IC50 = 78 nM T86591 C69PRB 90656440 IC50 = 42 nM T86591 C8C4XB 90656441 IC50 = 60 nM T86591 CA8C5T 90656442 IC50 = 386 nM T86591 C7DS4F 90656443 IC50 = 21 nM T86591 CUSA65 90656444 IC50 = 122 nM T86591 CUYO26 90656445 IC50 = 311 nM T86591 CXMC90 90676723 EC50 = 10000 nM T86591 CA9PL8 91663316 IC50 = 113 nM T86591 C7R6IK 101882290 EC50 > 10000 nM T86591 CCW4S0 101896435 EC50 = 210 nM T86591 CA6I4Y 101896436 EC50 = 3000 nM T86591 CFCE51 101896437 EC50 = 14400 nM T86591 C8CJR5 102004339 EC50 > 100000 nM T86591 C1CN0A 117629817 EC50 > 10000 nM T86591 C2NT4A 117940654 IC50 = 216 nM T86591 C8RZ0N 117940704 IC50 = 51 nM T86591 C2HMU9 117940709 IC50 = 433 nM T86591 C8M6VO 117940743 IC50 = 55 nM T86591 CAWZ74 117940820 IC50 = 23 nM T86591 C32XBP 117940859 IC50 = 569 nM T86591 C9BA5Q 117940874 IC50 = 80 nM T86591 CA95EY 117940949 IC50 = 66 nM T86591 CFYW64 117940962 IC50 = 608 nM T86591 C0J6WT 117940970 IC50 = 424 nM T86591 C0R8BX 117940999 IC50 = 56 nM T86591 CG7F5W 117941020 IC50 = 21 nM T86591 C3UR2N 117941053 IC50 = 678 nM T86591 C0VNL8 117941054 IC50 = 17 nM T86591 CWL20F 117941134 IC50 = 126 nM T86591 CHN6Z5 117941185 IC50 = 725 nM T86591 C4F1NK 117941228 IC50 = 420 nM T86591 C2B0NR 118708577 EC50 = 12000 nM T86591 CS9L7H 118708578 EC50 = 350 nM T86591 CVHW16 118708579 EC50 = 67 nM T86591 C1K9RV 118708580 EC50 = 70 nM T86591 CIU9H3 118708581 EC50 = 150 nM T86591 C1C6RK 118708582 EC50 = 240 nM T86591 CT4RD5 118714597 EC50 = 1300 nM T86591 C9M7RL 118714598 EC50 = 5800 nM T86591 C49HBU 118714599 EC50 = 3600 nM T86591 C5U4QT 118714600 EC50 = 19000 nM T86591 CN4PU6 118714603 EC50 = 2200 nM T86591 CA1RT3 118714624 EC50 = 4400 nM T86591 C8AS1X 118714625 EC50 = 5400 nM T86591 CB27OT 118714627 EC50 = 2900 nM T86591 C0X3NL 118714630 EC50 = 740 nM T86591 C7KS6D 118714631 EC50 = 9100 nM T86591 CR7I1H 118714632 EC50 = 4100 nM T86591 C0PTU8 118720593 EC50 = 4 nM T86591 CKC50A 118725345 EC50 = 18600 nM T86591 C5ENC7 118725346 EC50 = 5400 nM T86591 CTH73Y 118725347 EC50 = 5900 nM T86591 CQ4OY5 118725348 EC50 = 14400 nM T86591 C9M1BC 118725349 EC50 = 1300 nM T86591 CF3LH1 118726796 EC50 = 7750 nM T86591 C4URP2 118726797 EC50 = 5500 nM T86591 CNRJ62 118726798 EC50 = 7800 nM T86591 CSM7R4 118726800 EC50 = 7300 nM T86591 CG6Y7T 118726801 EC50 = 3800 nM T86591 C46WTE 118726802 EC50 = 3900 nM T86591 CSV2H4 118726804 EC50 = 4200 nM T86591 CJ2BR5 118726806 EC50 = 3800 nM T86591 C6YJQ9 118726808 EC50 = 6800 nM T86591 C2G5WT 118726809 EC50 = 2200 nM T86591 C92FYQ 118726811 EC50 = 1400 nM T86591 CC7A0V 118726812 EC50 = 5200 nM T86591 C4T1FZ 118726813 EC50 = 1200 nM T86591 C7UKX3 118726814 EC50 = 2100 nM T86591 C92IJW 118726815 EC50 = 220 nM T86591 COS6Z5 118727475 EC50 > 15000 nM T86591 C9OTJ4 118727476 EC50 > 15000 nM T86591 CC2JU8 118727477 EC50 = 3550 nM T86591 CUW31A 118727478 EC50 = 8100 nM T86591 CML56Z 118727479 IC50 > 10000 nM T86591 CF0YU2 118727480 IC50 > 10000 nM T86591 CI1H5O 118727481 IC50 = 1120 nM T86591 C5AO7P 118727482 EC50 = 2600 nM T86591 C8EC2D 118727483 EC50 = 10 nM T86591 C2F1AI 118727484 EC50 = 980 nM T86591 C4E3AX 121269371 EC50 = 6100 nM T86591 CW23RD 121269378 EC50 > 10000 nM T86591 C3AP2B 121269382 EC50 > 10000 nM T86591 CX4AN2 121269406 EC50 > 10000 nM T86591 CLRU83 121269424 EC50 > 10000 nM T86591 CC32JH 121277016 EC50 > 10000 nM T86591 C0BKL7 121277018 EC50 > 10000 nM T86591 CE3YL2 121277093 EC50 > 10000 nM T86591 CPA8J7 121277097 EC50 > 10000 nM T86591 C6TBD2 121345502 EC50 > 20000 nM T86591 C0BI8N 122183534 EC50 = 5900 nM T86591 CHYL24 122183546 EC50 = 19200 nM T86591 CBY0Q3 122184717 EC50 = 756 nM T86591 C9ZKJ7 122184718 EC50 > 100000 nM T86591 CX60IW 122184719 EC50 > 100000 nM T86591 CX8G2K 122184720 EC50 = 966 nM T86591 CQ6G2U 122184721 EC50 = 1922 nM T86591 C6EIX2 122184722 EC50 = 866 nM T86591 CTLQ94 122184723 EC50 = 981 nM T86591 CM1S7B 122370046 EC50 = 320 nM T86591 CT3O0F 122378601 EC50 = 3300 nM T86591 C7PMF2 122378603 EC50 = 760 nM T86591 CK6Q9P 122378605 EC50 = 800 nM T86591 CNY05V 122378606 EC50 = 28400 nM T86591 C9UB1X 125614030 EC50 = 1180 nM T86591 C3C9KP 125616706 EC50 = 830 nM T86591 C6ZHU9 125617607 EC50 = 970 nM T86591 C40QCP 125623112 EC50 = 770 nM T86591 C29TMV 127025858 EC50 = 17030 nM T86591 CB1UT6 127025866 EC50 = 4930 nM T86591 CQZB72 127025867 EC50 = 25410 nM T86591 C4-AUG-07 127027011 EC50 = 13210 nM T86591 C1I7VD 127027659 EC50 = 25210 nM T86591 C90UDI 127027730 EC50 = 30230 nM T86591 C2JP4N 127030270 IC50 = 800 nM T86591 CYAV89 127030271 IC50 = 8800 nM T86591 C5GVN3 127032266 IC50 = 6860 nM T86591 CA3L8P 127032267 IC50 = 850 nM T86591 C3WIN7 127033824 IC50 = 4600 nM T86591 C93YEH 127033825 IC50 = 680 nM T86591 C53RZG 127033833 IC50 = 108000 nM T86591 C0N5DO 127033834 IC50 = 4500 nM T86591 C0VMT1 127034100 IC50 = 820 nM T86591 CJ2QU3 127034101 IC50 = 650 nM T86591 CLBO13 127034102 IC50 = 7650 nM T86591 CQ49RY 127037376 EC50 = 90000 nM T86591 CMQ94Y 127037540 EC50 = 3800 nM T86591 C36UWM 127037541 EC50 = 103200 nM T86591 C82RIP 127042123 EC50 = 7000 nM T86591 C9H3DO 127042124 EC50 = 3000 nM T86591 C7J8AO 127042143 EC50 = 4000 nM T86591 C54WUI 127042144 EC50 = 900 nM T86591 C10ZDF 127042456 EC50 = 2000 nM T86591 C3PYC8 127043494 EC50 = 10.6 nM T86591 C19YRU 127043495 EC50 = 2.8 nM T86591 CP2GI3 127043496 EC50 = 2.3 nM T86591 C4EZC8 127043497 EC50 = 5.6 nM T86591 C1BI8N 127043498 EC50 = 6.8 nM T86591 C5WP3T 127043675 EC50 = 3.6 nM T86591 CQ72PD 127043676 EC50 = 4.3 nM T86591 CD0Q6O 127043844 EC50 = 2.7 nM T86591 CQ1O2V 127043845 EC50 > 2500 nM T86591 CIB59P 127043846 EC50 = 4 nM T86591 C5D7PK 127043847 EC50 = 3.4 nM T86591 CP83SU 127044158 EC50 = 94 nM T86591 C5YL1I 127044159 EC50 = 8.6 nM T86591 C3Z2WU 127044160 EC50 = 14.5 nM T86591 CZ2GY0 127044161 EC50 = 59 nM T86591 CLYV46 127044284 EC50 = 2.8 nM T86591 CG1RN9 127051847 EC50 = 2500 nM T86591 CL56FH 129147662 EC50 = 660 nM T86591 C1PGI4 132578432 EC50 = 210 nM T86591 C36ESP 132578434 EC50 = 150 nM T86591 C6W4KX 132578490 EC50 = 17 nM T86591 CX69BS 134139597 EC50 = 330 nM T86591 C0Y4CW 134154728 EC50 = 1000 nM T86591 CGX6K0 135444763 EC50 = 7500 nM T86591 CV6OP5 135513372 EC50 > 10000 nM T86591 CFT31G 135801082 EC50 = 12.1 nM T86591 CL6Q7I 136000613 EC50 = 10400 nM T86591 CYXD83 136036579 EC50 = 260 nM T86591 C9IU2J 136088972 IC50 = 100 nM T86591 CN7RH8 136264517 EC50 = 8.913 nM T86591 CW8QT1 137527725 IC50 > 80000 nM T86591 C7DS5O 137633219 EC50 = 1620 nM T86591 CYG4I2 137633420 EC50 = 2421 nM T86591 C15XNC 137637824 EC50 = 2824 nM T86591 CZT6M4 137637905 EC50 = 39 nM T86591 C6LI3N 137637955 EC50 = 764 nM T86591 C8FZ6W 137639177 EC50 = 5400 nM T86591 CI5ER2 137639724 EC50 = 2756 nM T86591 CKXQ78 137640612 EC50 = 42 nM T86591 CSP9K7 137641115 EC50 = 1250 nM T86591 CS82BE 137643489 EC50 > 5000 nM T86591 CCW0B2 137644269 EC50 > 5000 nM T86591 CBC61V 137647253 EC50 = 410 nM T86591 C93IRA 137648584 EC50 = 1164 nM T86591 CRB9Z7 137651528 EC50 = 1198 nM T86591 CHQ08L 137653711 EC50 = 46 nM T86591 CJ6DS1 137654442 EC50 = 1200 nM T86591 CS43WD 137654739 EC50 > 5000 nM T86591 CLA1N3 137655653 EC50 = 240 nM T86591 CZ84GI 137655707 EC50 = 1300 nM T86591 CQI07K 137656641 EC50 = 450 nM T86591 CGP3J1 137659100 EC50 = 100 nM T86591 CL1RG9 137659246 EC50 = 1963 nM T86591 COWM26 137659583 EC50 = 470 nM T86591 CUA42H 137660782 EC50 = 880 nM T86591 CC5X3V 139501076 EC50 = 25300 nM T86591 CFM9U6 139501078 EC50 = 5100 nM T86591 CHR98T 139501082 EC50 = 25600 nM T86591 C5WRM9 139501186 EC50 = 300 nM T86591 C9KYQ5 139501208 EC50 = 2100 nM T86591 CH3KJ0 139501210 EC50 = 8520 nM T86591 C35EGB 141511142 EC50 = 12690 nM T86591 C95BLC 141511161 EC50 = 11030 nM T86591 CZI51H 141511162 EC50 = 6990 nM T86591 CNUA15 141707372 EC50 = 1760 nM T86591 C7X1JD 141707373 EC50 > 2270 nM T86591 C9X1SL 141707374 EC50 = 1980 nM T86591 CI62UX 141707375 EC50 > 4010 nM T86591 C9GMY6 141707376 EC50 = 2410 nM T86591 C2JZW1 141707377 EC50 > 1340 nM T86591 C8ZQX0 141707379 EC50 = 1230 nM T86591 CP5N7E 141707380 EC50 > 2740 nM T86591 CH60ZV 141707382 EC50 = 1390 nM T86591 CKS10N 145704693 EC50 = 430 nM T86591 CT73UW 145949449 EC50 > 10000 nM T86591 COKZ54 145949774 EC50 = 10000 nM T86591 C04TKM 145949801 EC50 = 10000 nM T86591 CLS49D 145950904 EC50 = 10000 nM T86591 CT5BL8 145951025 EC50 > 10000 nM T86591 CGE1B3 145951206 EC50 > 10000 nM T86591 CQ6N2Z 145951479 EC50 > 10000 nM T86591 CI08MP 145951689 EC50 > 10000 nM T86591 C4GBZ5 145951912 EC50 = 2000 nM T86591 CURD19 145952141 EC50 = 300 nM T86591 C9AST8 145952202 EC50 > 10000 nM T86591 C85OUK 145952859 EC50 > 10000 nM T86591 CQGS02 145953624 EC50 = 10000 nM T86591 C96FER 145954306 EC50 > 10000 nM T86591 CV6L7A 145954353 EC50 > 10000 nM T86591 CQ93BF 145954620 EC50 > 10000 nM T86591 CT0HJ3 145955210 EC50 > 10000 nM T86591 C0NLP6 145955315 EC50 > 10000 nM T86591 CLW25D 145955603 EC50 > 10000 nM T86591 CI4K0Z 145955653 EC50 > 10000 nM T86591 CD3E4U 145955709 EC50 = 1000 nM T86591 C5X9NS 145956690 EC50 = 10000 nM T86591 C8X9ZN 145956749 EC50 > 10000 nM T86591 CL0C9N 145956984 EC50 > 10000 nM T86591 CS1W8N 145957036 EC50 > 10000 nM T86591 C4C3IO 145957135 EC50 = 10000 nM T86591 CJA0E5 145957371 EC50 = 10000 nM T86591 CTIJ56 145957793 EC50 = 10000 nM T86591 CCW82O 145958068 EC50 = 10000 nM T86591 CZ7X5B 145958164 EC50 = 1000 nM T86591 CXR2V7 145959160 EC50 > 10000 nM T86591 CA01SL 145959379 EC50 > 10000 nM T86591 C9VHW3 145959494 EC50 > 10000 nM T86591 C08RPJ 145959499 EC50 = 10000 nM T86591 CCR02D 145959510 EC50 = 10000 nM T86591 CR54HC 145959653 EC50 = 10000 nM T86591 CNH07S 145960072 EC50 > 10000 nM T86591 C28YLS 145960168 EC50 > 10000 nM T86591 CHL06X 145960211 EC50 > 10000 nM T86591 CCF02H 145964530 IC50 = 8000 nM T86591 C56SHA 145964597 IC50 = 3500 nM T86591 C5DH4X 145964745 EC50 > 10000 nM T86591 C5H8EZ 145965425 IC50 = 1900 nM T86591 CT8AU9 145971273 EC50 > 10000 nM T86591 C9GPT8 145972429 EC50 > 10000 nM T86591 CA0RD6 145973168 EC50 > 10000 nM T86591 C0LTV9 145973176 EC50 > 10000 nM T86591 CJDH32 145975435 EC50 > 10000 nM T86591 C98CHS 145977976 IC50 = 6600 nM T86591 C0KP3F 145980573 EC50 > 10000 nM T86591 C1Q6PV 145980608 EC50 = 7310 nM T86591 CKR43C 145981599 EC50 > 10000 nM T86591 C87UAM 145982210 EC50 = 5260 nM T86591 CFY8U2 145982433 EC50 > 10000 nM T86591 C4D7TZ 145982651 EC50 > 10000 nM T86591 CT0YS3 145982746 EC50 > 10000 nM T86591 C65PGI 145982771 EC50 > 10000 nM T86591 CTFM01 145982798 EC50 > 10000 nM T86591 C65FME 145983252 EC50 > 10000 nM T86591 CH1XJ8 145983321 EC50 > 10000 nM T86591 C3WJZ8 145983637 EC50 > 10000 nM T86591 CP4W3R 145983705 EC50 > 10000 nM T86591 CT90OW 145983779 EC50 > 10000 nM T86591 CFJ94I 145984084 EC50 > 10000 nM T86591 CH9MK6 145984248 EC50 = 9500 nM T86591 C8V7OD 145984577 EC50 > 10000 nM T86591 C4LN8E 145984731 EC50 > 10000 nM T86591 CIV2P1 145984795 EC50 > 10000 nM T86591 C0C2SU 145984820 EC50 > 10000 nM T86591 CQ1TB7 145984906 EC50 > 10000 nM T86591 CV84PQ 145985229 EC50 > 10000 nM T86591 CH9OI0 145985286 EC50 > 10000 nM T86591 CG8R3L 145985481 EC50 > 10000 nM T86591 C9LA1O 145985668 EC50 > 10000 nM T86591 CB47FE 145985838 EC50 = 5900 nM T86591 CRAK83 145985994 EC50 > 10000 nM T86591 CMAN27 145986012 EC50 = 27000 nM T86591 CA8JQ5 145986026 EC50 = 2600 nM T86591 CAE95K 145986458 EC50 > 10000 nM T86591 CW7Y4G 145986696 EC50 > 10000 nM T86591 CBOR53 145986704 EC50 > 10000 nM T86591 C0G2WE 145988431 EC50 > 10000 nM T86591 C75DSN 145989198 EC50 > 10000 nM T86591 CI39OJ 145989913 EC50 > 10000 nM T86591 CJ76KD 145990303 EC50 > 10000 nM T86591 CV2FB6 145992078 EC50 > 10000 nM T86591 C6F0LJ 145992170 EC50 > 10000 nM T86591 CP79UQ 145992176 EC50 > 10000 nM T86591 CCV39B 145994196 EC50 > 10000 nM T86591 C0O2PY 146036004 EC50 = 1530 nM T86591 C0PRO4 151689224 EC50 = 1800 nM T86591 C7X3AL 153763221 EC50 = 5200 nM T86591 C2L3TU 155510528 EC50 = 460 nM T86591 CD5QM6 155511861 EC50 = 27 nM T86591 CJRW35 155512467 IC50 = 18 nM T86591 CJ69KC 155512807 EC50 = 31 nM T86591 CCGW81 155512868 EC50 = 2200 nM T86591 CUNF95 155513665 EC50 = 21000 nM T86591 C3Z6VL 155514089 EC50 = 26000 nM T86591 CDA4C9 155515667 IC50 = 12900 nM T86591 CICX19 155516325 EC50 = 3100 nM T86591 C43TAC 155516878 EC50 = 960 nM T86591 C9NPC1 155517336 EC50 = 5000 nM T86591 CS48YI 155517472 EC50 = 100 nM T86591 C2COG3 155517895 EC50 = 2300 nM T86591 C2C4OZ 155518329 EC50 = 1400 nM T86591 C1POU5 155518522 EC50 = 3100 nM T86591 CVAX73 155519415 EC50 = 52 nM T86591 CB68OA 155520333 EC50 = 900 nM T86591 C86OCS 155520630 IC50 = 33 nM T86591 C6R1TF 155520683 EC50 = 250 nM T86591 C6EW5F 155523441 EC50 = 810 nM T86591 C3GH8U 155523815 EC50 = 580 nM T86591 C4Q7TF 155524299 EC50 = 100 nM T86591 C9ED1Q 155524951 EC50 = 29 nM T86591 CX5GA6 155525020 EC50 = 18 nM T86591 CS9N2M 155525414 EC50 = 680 nM T86591 C4GEH1 155525496 IC50 = 38140 nM T86591 CV51OZ 155526003 IC50 = 23120 nM T86591 C95KYP 155526365 EC50 = 1800 nM T86591 CSJ48X 155527435 EC50 = 3423 nM T86591 CS3J1W 155527996 EC50 = 4000 nM T86591 CO7NR2 155528574 EC50 = 2600 nM T86591 C3LZQ1 155528955 EC50 = 510 nM T86591 CJNU21 155529721 EC50 = 37 nM T86591 C9YTH8 155530420 EC50 = 400 nM T86591 COG5A0 155530735 EC50 = 25000 nM T86591 CQ1H7L 155531716 EC50 = 67 nM T86591 C6W2JV 155531862 EC50 = 540 nM T86591 C4YW2E 155532130 EC50 = 1616 nM T86591 C2O9VS 155532185 EC50 = 500 nM T86591 C08UVN 155532889 EC50 = 810 nM T86591 CBH5U3 155533072 EC50 = 360 nM T86591 C63HSA 155534748 EC50 = 8 nM T86591 CK89PE 155534755 EC50 = 47000 nM T86591 CE7I8Q 155534885 EC50 = 18000 nM T86591 CC9T6U 155535078 EC50 = 1450 nM T86591 C2FU1O 155535195 IC50 = 122 nM T86591 C0B5MT 155535253 EC50 = 250 nM T86591 CS86YB 155535303 EC50 = 380 nM T86591 C8EQI9 155536324 EC50 = 1450 nM T86591 CR9BE4 155536793 IC50 = 31440 nM T86591 CHC04X 155536991 EC50 = 700 nM T86591 CN48LF 155537424 EC50 = 130 nM T86591 CM7S9F 155537835 IC50 = 89300 nM T86591 CE2LR1 155538630 EC50 = 1120 nM T86591 CLE42C 155538881 EC50 = 1610 nM T86591 C3R9YL 155539254 EC50 = 20000 nM T86591 C4KMH1 155540131 EC50 = 385 nM T86591 CJC0K1 155540534 EC50 = 1900 nM T86591 CVL59Z 155540834 EC50 = 8974 nM T86591 CP3I4H 155541634 EC50 = 11000 nM T86591 C64FRG 155541703 IC50 = 1100 nM T86591 CSI9G7 155541727 EC50 = 770 nM T86591 CJB39Q 155541750 EC50 = 1000 nM T86591 C19LXF 155543073 EC50 = 1240 nM T86591 CXI91F 155543520 IC50 = 394 nM T86591 C8MEV9 155543569 EC50 = 2821 nM T86591 C1YSQ7 155545016 EC50 = 33 nM T86591 C5Q6WG 155545482 EC50 = 1360 nM T86591 CLH91J 155545920 IC50 = 32 nM T86591 CNSF75 155546388 IC50 = 30990 nM T86591 CFQ28J 155546921 EC50 = 1900 nM T86591 C0A1VM 155547028 EC50 > 3570 nM T86591 C0H7JO 155547646 EC50 = 1000 nM T86591 C2QGR5 155549327 EC50 = 5400 nM T86591 C4E8HZ 155550405 EC50 = 56 nM T86591 CZ59YK 155550531 IC50 = 18 nM T86591 C87TQJ 155551096 EC50 = 4000 nM T86591 C2MTF9 155552428 EC50 = 3800 nM T86591 CWG10F 155552953 IC50 = 11440 nM T86591 C3KD0I 155553701 IC50 = 1240 nM T86591 C7IN4B 155554421 EC50 = 1400 nM T86591 CSG9P5 155555340 EC50 = 27 nM T86591 CJQ54R 155556924 EC50 = 7500 nM T86591 CN4ZU8 155558177 EC50 = 740 nM T86591 CEI8F1 155558276 EC50 = 4400 nM T86591 CM52UW 155560868 EC50 = 1200 nM T86591 CUDT29 155561763 IC50 = 200 nM T86591 C3DN4K 155562634 EC50 = 900 nM T86591 CK94IU 155564010 IC50 = 5040 nM T86591 CG02XL 155565451 EC50 > 10000 nM T86591 CG57AR 155566529 EC50 = 10000 nM T86591 C3FK2M 155566781 EC50 = 1000 nM T86591 CO07PA 155568591 EC50 = 930 nM T86591 CPWE70 155569128 EC50 = 40 nM T86591 CQP4Y0 155569313 EC50 = 2400 nM T86591 C26RKO 155569383 EC50 = 1450 nM T86591 CI24DH 155569680 EC50 = 184 nM T86591 D00TFA 3392731 Ki = 0.0541 nM T86591 D01POG 657048 EC50 < 20 nM T86591 D01RPM 11645581 IC50 > 15000 nM T86591 D02TRN 445638 IC50 = 1700 nM T86591 D02TVS 985 IC50 = 1500 nM T86591 D02WFA 5281 IC50 = 1100 nM T86591 D03LOG 5280450 IC50 = 1100 nM T86591 D04DYM 6518171 EC50 = 55300 nM T86591 D04FVX 44220886 IC50 > 15000 nM T86591 D05CLM 9870304 EC50 = 6 nM T86591 D06GYO 5282316 IC50 = 9600 nM T86591 D06IHG 24836820 IC50 > 15000 nM T86591 D06MDX 11483970 EC50 = 190 nM T86591 D06NHI 9843045 EC50 = 740 nM T86591 D06RRD 2797 EC50 = 39600 nM T86591 D06TXM 24816385 EC50 = 1000 nM T86591 D06VBQ 46233311 IC50 > 10000 nM T86591 D07LUJ 64945 EC50 = 41310 nM T86591 D07MBC 5283454 EC50 = 110 nM T86591 D08JHR 16103199 EC50 > 10000000 nM T86591 D08OBF 11005 IC50 = 5400 nM T86591 D08QKF 9954280 IC50 > 15000 nM T86591 D08QXD 9935197 EC50 = 125 nM T86591 D08UWZ 16725047 EC50 = 9.6 nM T86591 D08WRU 16103197 EC50 = 100 nM T86591 D08ZYC 11595431 Ki < 3162.28 nM T86591 D09JII 9891946 EC50 = 4.1 nM T86591 D09XCX 5694 EC50 = 130 nM T86591 D0A4EA 445639 IC50 = 600 nM T86591 D0C5SV 5280934 IC50 = 1200 nM T86591 D0E7NO 2969 IC50 = 30000 nM T86591 D0F0MP 9889841 EC50 = 247 nM T86591 D0H4US 11149906 EC50 = 700 nM T86591 D0HD9P 444899 IC50 = 1200 nM T86591 D0J3UU 11460087 EC50 = 3890.45 nM T86591 D0K1TQ 9934458 EC50 = 920 nM T86591 D0M9LL 44221100 IC50 = 1600 nM T86591 D0N0UC 3893 IC50 = 30000 nM T86591 D0NM0G 2800647 IC50 > 10000 nM T86591 D0O2US 9870584 Ki = 1100 nM T86591 D0P5QM 44221101 IC50 = 1100 nM T86591 D0Q4UD 44220888 IC50 > 15000 nM T86591 D0W7RI 5311242 EC50 = 340 nM T86591 D0W9WU 44220887 IC50 > 15000 nM T86591 D0XR8Q 1517 EC50 = 170 nM T86591 D0YK9T 6603901 EC50 = 977 nM T86591 D0Z4NW 44220889 IC50 > 15000 nM T86591 D0Z7OX 9890319 EC50 = 149.5 nM T69494 D00ENY 33032 IC50 = 70 nM T69494 D01JEU 4054 Ki = 540 nM T69494 D01ZII 2726 IC50 = 600 nM T69494 D02KRS 2130 Ki = 10500 nM T69494 D09OBB 5360696 Ki = 1680 nM T69494 D0D9FV 4601 Ki = 6000 nM T69494 D0R1WR 4919 Ki = 1700 nM T69494 D0RM9Q 68778 Ki = 11700 nM T69494 D0T3HY 5359272 IC50 = 2500 nM T69494 D0UM7O 3821 Ki = 420 nM T69494 D02VKC 3272524 IC50 > 100000 nM T69494 D04WUA 219101 IC50 = 7 nM T69494 D09BEG 192711 Ki = 1.94 nM T69494 D0B0NQ 127894 IC50 = 12100 nM T69494 D0LI1C 44469321 IC50 > 10000 nM T69494 D0N1HW 5311200 Ki > 10000 nM T69494 D0N3EJ 10200813 IC50 = 6 nM T69494 D00MFY 108099 IC50 = 976 nM T69494 D02KLW 180081 Ki = 1.2 nM T69494 D03HDP 9816526 IC50 = 4677351.41 nM T69494 D03RZU 9842186 Ki = 179 nM T69494 D06DLQ 5950212 IC50 = 18 nM T69494 D06RCS 156328 IC50 = 4 nM T69494 D09CKF 5486198 IC50 = 5.9 nM T69494 D0H1FV 68736 IC50 = 54 nM T69494 D0K0DB 6604887 Ki = 5.6 nM T69494 D0O4JH 9816093 IC50 = 29 nM T69494 CYCS18 3008 IC50 = 240 nM T69494 CE41ZK 7594 IC50 = 3450 nM T69494 CTC8N0 14657 IC50 > 100000 nM T69494 CJZ59G 19476 Ki = 21700 nM T69494 CNS2V1 19478 Ki = 20800 nM T69494 C5EO7I 22648 IC50 = 1600 nM T69494 CKO78N 27491 IC50 = 9800 nM T69494 CM4VK9 33142 IC50 = 6800 nM T69494 C4CP3H 35998 Ki = 9500 nM T69494 CO6M2K 41011 IC50 = 13300 nM T69494 CAN7Z1 64245 Ki = 3800 nM T69494 CV3PD7 64352 Ki = 600 nM T69494 C8CZ1E 64600 IC50 > 10000 nM T69494 CL7AZ0 86625 Ki = 33300 nM T69494 CY65GC 112416 IC50 > 10000 nM T69494 CLK95E 177328 IC50 = 8 nM T69494 CDM25N 230867 IC50 > 10000 nM T69494 C40JGX 247670 IC50 = 3300 nM T69494 C0PUC2 344343 IC50 = 134 nM T69494 CIX84S 407725 IC50 > 10000 nM T69494 CCO6D8 428911 IC50 > 10000 nM T69494 CROX25 480185 IC50 = 1190 nM T69494 CI2DZ9 613780 IC50 = 17000 nM T69494 C6R7DK 617841 IC50 = 1000 nM T69494 C7JED1 655777 IC50 = 2100 nM T69494 CQD2N8 728567 IC50 > 10000 nM T69494 C9O3DA 3010129 Ki = 15200 nM T69494 C32DCS 3018579 IC50 = 460 nM T69494 CCW10K 3035668 IC50 = 5000 nM T69494 C9LN3O 3072821 IC50 = 264 nM T69494 COF48J 3246533 IC50 = 639 nM T69494 C6G4UP 3315413 IC50 > 10000 nM T69494 C5OHM8 3481675 IC50 > 100000 nM T69494 CZF7B5 5026275 Ki = 6943 nM T69494 CI8JG6 5100144 Ki = 7210 nM T69494 C9RQU0 5276622 Ki = 1610 nM T69494 CE3U5V 5276624 Ki = 4440 nM T69494 CU9Y4H 5276625 Ki = 1720 nM T69494 CZWX37 5360697 Ki = 220 nM T69494 CX1KW7 6603754 IC50 = 86 nM T69494 C9C8BQ 6604117 Ki = 13 nM T69494 CB50FH 6604872 IC50 > 10000 nM T69494 CIS53Q 6918409 IC50 = 4 nM T69494 CP3QT1 9560223 IC50 = 32359.37 nM T69494 CPO03K 9797767 IC50 = 12 nM T69494 CX3U7N 9813501 Ki = 8 nM T69494 CJM0W8 9816863 Ki = 2 nM T69494 C2FVL8 9818804 IC50 > 10000 nM T69494 CP9QV1 9838551 IC50 = 148 nM T69494 CB31LS 9855978 Ki = 3 nM T69494 CTUM52 9856417 Ki = 4 nM T69494 CS3C1T 9863233 IC50 = 6 nM T69494 C8DN6M 9868551 IC50 = 8 nM T69494 CYSB08 9878065 Ki = 5 nM T69494 CV1P8X 9902229 IC50 = 18 nM T69494 CHV52Y 9902230 IC50 = 31 nM T69494 C6GCF5 9903013 IC50 = 19 nM T69494 C72EDR 9905123 Ki = 3.5 nM T69494 CUN81Q 9905249 Ki > 10000 nM T69494 C9XIG6 9919363 IC50 = 240 nM T69494 CQ3L1X 9921302 Ki = 3 nM T69494 CJ46NU 9921303 Ki = 8 nM T69494 CBE1Y9 9921863 Ki = 4 nM T69494 C5E7KC 9943680 Ki = 8 nM T69494 COZF94 9964271 IC50 = 1600 nM T69494 C4I7UJ 9964754 Ki = 4 nM T69494 CMI27N 9968278 IC50 = 106 nM T69494 C2K7RI 9998705 Ki = 7 nM T69494 C3G9NW 10013264 Ki = 190 nM T69494 CV7R9F 10020040 Ki > 10000 nM T69494 CV5KA9 10040420 IC50 = 8.7 nM T69494 CB8KW6 10048025 IC50 > 10000 nM T69494 C30CGH 10058555 IC50 = 10000 nM T69494 CI1U0P 10103573 IC50 = 2300 nM T69494 C2HX7F 10106426 IC50 = 45 nM T69494 CVP15K 10132591 IC50 = 47 nM T69494 CHB56O 10134304 IC50 = 8 nM T69494 CT93DE 10135057 IC50 = 54 nM T69494 CCG86J 10136334 IC50 = 17 nM T69494 C62KMH 10157570 IC50 = 5 nM T69494 CAG04L 10177679 IC50 = 4 nM T69494 CJ14NF 10178824 IC50 = 17 nM T69494 C9UFL7 10179770 IC50 = 131 nM T69494 CJ86CV 10201898 IC50 = 26 nM T69494 C92NFX 10220703 Ki = 4080 nM T69494 C3NB6R 10242135 Ki = 790 nM T69494 C8R2AC 10243335 IC50 = 370 nM T69494 C4M9CI 10263627 IC50 = 95 nM T69494 CH31DX 10267394 Ki > 10000 nM T69494 CIVO90 10273343 IC50 = 40 nM T69494 CK7VD6 10290921 IC50 = 16 nM T69494 CU89JD 10314060 Ki > 10000 nM T69494 C3YU6I 10331572 IC50 = 470 nM T69494 CLS1Y9 10342393 Ki > 10000 nM T69494 C9AJ7X 10378304 IC50 = 82 nM T69494 C58HNW 10473406 Ki = 4.9 nM T69494 C2J1PI 10475669 IC50 = 139 nM T69494 CG2HA7 10497882 Ki = 260 nM T69494 C0KB1F 10497883 Ki = 2600 nM T69494 C7W9LB 10498834 IC50 = 59 nM T69494 CY91ED 10498835 Ki = 110 nM T69494 CZ6J9T 10512659 IC50 = 780 nM T69494 CQNE23 10514172 IC50 = 11000 nM T69494 C71UOL 10546555 Ki = 2700 nM T69494 CHWQ56 10550344 Ki > 10000 nM T69494 CG6P3E 10552301 Ki > 10000 nM T69494 CA3S6R 10561180 IC50 = 151356124.8 nM T69494 CYX93H 10562939 IC50 > 100000 nM T69494 C1H6ZO 10594610 IC50 = 4000 nM T69494 CN5G4K 10609584 IC50 = 2800 nM T69494 C7WKJ2 10610792 IC50 > 100000 nM T69494 CGR5I2 10611559 IC50 = 160 nM T69494 C72ELH 10615770 IC50 = 196 nM T69494 C6CX0R 10617348 Ki = 720 nM T69494 C4Z7OP 10617349 Ki = 2200 nM T69494 C3R8ML 10618320 Ki = 22000 nM T69494 C7NBC4 10632607 IC50 = 1800 nM T69494 CE3TG4 10638058 IC50 = 640 nM T69494 CB7QK1 10638963 IC50 = 82 nM T69494 C0O6ZI 10658567 IC50 > 100000 nM T69494 C34MOV 10665363 Ki = 6700 nM T69494 C21KCF 10666040 Ki = 380 nM T69494 CUFJ06 10682422 IC50 = 1900 nM T69494 C24OBP 10683434 IC50 = 28840315.03 nM T69494 CY9A6G 10689687 IC50 = 240 nM T69494 COH5Y4 10705621 IC50 = 3100 nM T69494 CZS7N2 10707059 IC50 = 3600 nM T69494 C54SKU 10707115 IC50 = 130 nM T69494 CG5L3V 10717311 Ki > 10000 nM T69494 C8XC0W 10719152 Ki > 10000 nM T69494 CR4D3C 10719153 Ki > 10000 nM T69494 CE1F8Z 10726784 IC50 = 15000 nM T69494 C9BV5R 10729534 IC50 > 100000 nM T69494 CB2L8N 10742982 Ki > 10000 nM T69494 CA12MI 10751444 IC50 = 9300 nM T69494 CIW54Y 10752476 IC50 > 100000 nM T69494 CB10GW 10774166 IC50 = 10000000 nM T69494 C09IND 10783593 Ki = 11000 nM T69494 C6UDT4 10783594 Ki = 5800 nM T69494 CO40KL 10784562 Ki = 60 nM T69494 C9H0TI 10800053 IC50 > 100000 nM T69494 CT09ZK 10822409 IC50 = 16000 nM T69494 C1GPC8 10823051 IC50 = 1400 nM T69494 C82SBI 10823505 IC50 = 630957344.5 nM T69494 C3B9HI 10823814 IC50 > 100000 nM T69494 C27OLZ 10824301 IC50 = 73 nM T69494 C02QUD 10824747 IC50 > 100000 nM T69494 CQAK84 10831541 Ki = 920 nM T69494 CC07RZ 10836171 Ki > 10000 nM T69494 CTO97D 10845927 IC50 = 10000000 nM T69494 CY7F4U 10849759 IC50 = 150 nM T69494 CI64CK 10851503 IC50 = 4300 nM T69494 C4HR7X 10884456 Ki > 10000 nM T69494 C1Y9ID 10971999 Ki > 10000 nM T69494 CJOC58 11048224 Ki > 10000 nM T69494 CM65YK 11069974 Ki > 10000 nM T69494 C6P7AB 11218368 Ki = 1700 nM T69494 C2C5BR 11747939 IC50 = 53000 nM T69494 CXLW54 11948707 Ki > 10000 nM T69494 C0W8NV 12150769 IC50 = 61000 nM T69494 C3E7QH 12628908 IC50 > 10000 nM T69494 COST51 13477634 IC50 = 112000 nM T69494 CYV6B5 13781931 IC50 = 358 nM T69494 C2SEG3 13781932 IC50 = 32000 nM T69494 CG08MN 13781936 IC50 = 275 nM T69494 C3FCB2 13781939 IC50 = 38300 nM T69494 CM7J6R 13975369 IC50 = 26915.35 nM T69494 CX20PD 14125583 IC50 > 10000 nM T69494 CJNM56 14292033 IC50 = 4350 nM T69494 CRJ0L3 14771666 IC50 = 498 nM T69494 CE0KP4 14771667 IC50 = 1570 nM T69494 CM29BA 14771668 IC50 = 2110 nM T69494 C5SU1R 14771669 IC50 = 1100 nM T69494 CWMO41 14771670 IC50 = 4150 nM T69494 CPB79U 14771672 IC50 = 34000 nM T69494 C7M1AK 14771673 IC50 > 10000 nM T69494 CTBR56 14771675 IC50 > 10000 nM T69494 CQ1ZC3 14771677 IC50 = 5000 nM T69494 CX4H7W 14771682 IC50 = 49000 nM T69494 CIY37H 14771684 IC50 = 2050 nM T69494 CP4LQ5 14771685 IC50 = 5700 nM T69494 CR67MN 14771686 IC50 = 1900 nM T69494 CEQV06 14771688 IC50 = 12000 nM T69494 CH2R4M 14771689 IC50 = 4300 nM T69494 CDHN24 14771691 IC50 > 10000 nM T69494 C3WK2C 14771692 IC50 > 10000 nM T69494 CJ21YE 14771693 IC50 > 10000 nM T69494 CJY5N0 14771694 IC50 = 10000 nM T69494 C2NW9K 14771695 IC50 > 10000 nM T69494 C47EWB 14771696 IC50 = 32000 nM T69494 CF6OB9 14771697 IC50 > 10000 nM T69494 CRK3S4 14771698 IC50 > 10000 nM T69494 CO4Z3M 14771699 IC50 > 10000 nM T69494 C6A4YT 14771702 IC50 > 10000 nM T69494 CS9Z3L 14771705 IC50 = 5000 nM T69494 C8S0BC 14771707 IC50 = 2500 nM T69494 CU94AL 14771709 IC50 > 10000 nM T69494 C2FO3S 14771711 IC50 = 2000 nM T69494 CF2L5J 14771713 IC50 = 4000 nM T69494 CL0GD1 14771715 IC50 > 10000 nM T69494 C8B9LE 14771717 IC50 > 10000 nM T69494 CGJB25 14771719 IC50 = 3500 nM T69494 C6JM8H 14771721 IC50 > 10000 nM T69494 C0BZJ6 14771723 IC50 > 10000 nM T69494 CCW53V 14771725 IC50 > 10000 nM T69494 CCMA03 14771728 IC50 = 37000 nM T69494 CXGT50 14771729 IC50 > 10000 nM T69494 CZSE76 14771731 IC50 > 100000 nM T69494 CCZ3L7 14771734 IC50 > 10000 nM T69494 CL7NO6 14771736 IC50 > 10000 nM T69494 C64VXZ 14771738 IC50 > 10000 nM T69494 CQ92IT 14771742 IC50 > 9600 nM T69494 C53BMJ 14771744 IC50 > 10000 nM T69494 CR78EM 14877965 IC50 = 16300 nM T69494 CJWC98 14877967 IC50 = 781 nM T69494 C8L6WJ 15113312 Ki = 3042 nM T69494 CEOS76 15523910 Ki = 7.5 nM T69494 CIW1V2 15870643 IC50 = 1.5 nM T69494 CY4QO6 15917395 Ki = 17400 nM T69494 C6D2LG 16110277 IC50 = 359 nM T69494 C7NYH8 16110280 IC50 = 380 nM T69494 CZ2IS9 16660294 Ki > 10000 nM T69494 CH1U7N 16783390 Ki = 380 nM T69494 C4BCD0 16784177 Ki = 1100 nM T69494 CKEF25 19785444 IC50 = 170 nM T69494 C6HVQ3 19785447 IC50 = 480 nM T69494 CC0J8U 19785449 IC50 = 6400 nM T69494 CN8XP4 19785450 IC50 = 680 nM T69494 COD2C1 19785452 IC50 = 370 nM T69494 C7T8JC 19958494 Ki > 10000 nM T69494 C6LI5E 19958507 Ki > 10000 nM T69494 C7MUY5 20666336 IC50 = 17000 nM T69494 CW0AT1 21189968 IC50 = 724435960.1 nM T69494 CE3OI8 21396684 IC50 = 7079.46 nM T69494 CBN84K 22065997 Ki > 10000 nM T69494 C9Q5AO 22605919 Ki = 380 nM T69494 CAH62L 22605921 Ki = 110 nM T69494 C6H0QC 22605923 Ki = 190 nM T69494 CW3JL4 22605927 Ki = 380 nM T69494 CT0PV3 22605938 Ki = 150 nM T69494 C9D5AR 25211257 IC50 = 60000 nM T69494 C1MWY0 44118332 IC50 = 154881.66 nM T69494 C0J2GB 44118333 IC50 = 77624.71 nM T69494 CNK26P 44250141 IC50 = 370000 nM T69494 CC32QT 44268120 IC50 = 27 nM T69494 C5P8RI 44268131 IC50 = 130 nM T69494 CW4XE5 44268133 IC50 = 0.8 nM T69494 C7STQ5 44268139 IC50 = 38 nM T69494 CG6T3J 44268140 IC50 = 7.4 nM T69494 C1DHG0 44268169 IC50 = 250 nM T69494 C4W0VD 44268176 IC50 = 860 nM T69494 CCS1V3 44268177 IC50 = 1100 nM T69494 C0KC1V 44268182 IC50 = 370 nM T69494 CUF3D9 44268187 IC50 = 1.2 nM T69494 CL67WI 44268196 IC50 = 120 nM T69494 CN71DL 44268201 IC50 = 31 nM T69494 CVN1B5 44268208 IC50 = 8.1 nM T69494 CC5KV6 44268212 IC50 = 0.5 nM T69494 C2L8JR 44268217 IC50 = 1 nM T69494 CXP56A 44268218 IC50 = 1.7 nM T69494 CC3UJ9 44268225 IC50 = 160 nM T69494 C3FJ0O 44268282 IC50 = 1.5 nM T69494 C7ALC5 44268285 IC50 = 17 nM T69494 CRT6N1 44268299 IC50 = 9.7 nM T69494 CC2OD4 44278111 Ki > 10000 nM T69494 CRMA84 44278114 Ki > 10000 nM T69494 CF0Y4M 44278115 Ki > 10000 nM T69494 C3FO8X 44288293 IC50 = 64 nM T69494 CI0ZP9 44288318 IC50 = 1000 nM T69494 C8GQ4A 44304811 IC50 = 26400 nM T69494 CQRK31 44309145 Ki = 3.8 nM T69494 CHYZ41 44309146 Ki = 3.4 nM T69494 CU2Z3N 44309182 Ki = 11.3 nM T69494 CB18TU 44309199 Ki = 7.5 nM T69494 CMJV60 44309200 Ki = 15 nM T69494 C8UR6M 44309202 Ki = 22.6 nM T69494 CK26BL 44309367 Ki = 3.8 nM T69494 C8Y5ZU 44309368 Ki = 22.6 nM T69494 CHC12P 44309385 Ki = 19.9 nM T69494 C9Y7AI 44309455 Ki = 2230 nM T69494 CCQN61 44309978 Ki = 8300 nM T69494 C4UZG0 44309993 Ki > 10000 nM T69494 CLYS40 44309995 Ki = 4400 nM T69494 CU0EA9 44310036 Ki = 100000 nM T69494 C7M5HP 44310050 Ki = 2030 nM T69494 C09JTN 44310052 Ki > 10000 nM T69494 C4MD0R 44310071 Ki = 12000 nM T69494 CY6O4H 44310073 Ki > 10000 nM T69494 CD5R0G 44318068 IC50 > 10000 nM T69494 C9UI8D 44318072 IC50 > 10000 nM T69494 C2H6BO 44328124 Ki > 10000 nM T69494 CFTP16 44328133 Ki > 10000 nM T69494 CW97OV 44328157 Ki > 10000 nM T69494 C1H2OZ 44328180 Ki > 10000 nM T69494 C43OCF 44338473 IC50 = 555 nM T69494 C1X2AG 44338533 IC50 = 6458 nM T69494 C9J4ME 44348419 IC50 = 120 nM T69494 C8BJP5 44352415 Ki = 4100 nM T69494 C6OZ2G 44354079 IC50 = 150 nM T69494 CYCL52 44354092 IC50 = 100 nM T69494 CK8TF1 44354093 IC50 = 150 nM T69494 CG2NB1 44354094 IC50 = 130 nM T69494 CCZ3M6 44355999 IC50 > 20000 nM T69494 CCN4L7 44356001 IC50 = 8480 nM T69494 CCHL41 44356109 IC50 = 23 nM T69494 CVN1P8 44356169 IC50 = 125 nM T69494 CDK3U7 44356310 IC50 = 69 nM T69494 CCDZ62 44362569 IC50 = 1601 nM T69494 C6LI1X 44362599 IC50 = 925 nM T69494 CD2M5S 44362600 IC50 = 685 nM T69494 C4B8XA 44362879 IC50 = 1670 nM T69494 CK8I1S 44362880 IC50 > 10000 nM T69494 CM10AB 44362916 IC50 > 10000 nM T69494 C0UD7R 44364816 Ki = 6587 nM T69494 C6PYE7 44379376 IC50 = 360 nM T69494 CQ5M0E 44380397 Ki = 260 nM T69494 C7YA9Q 44380479 Ki = 1100 nM T69494 C6FJW1 44380593 Ki = 15000 nM T69494 CGCB36 44380594 Ki = 7500 nM T69494 CG85AM 44380820 Ki = 9 nM T69494 CP76NX 44380878 Ki = 750 nM T69494 C9FWX4 44393025 IC50 = 17 nM T69494 CF6X3K 44460274 IC50 > 10000 nM T69494 CZS51T 44460446 IC50 > 10000 nM T69494 CNHZ76 45259280 IC50 = 65 nM T69494 C8N5JV 45259282 IC50 = 60 nM T69494 CW90NX 45259285 IC50 = 40 nM T69494 CTQP21 45259290 IC50 = 3 nM T69494 CN0MX8 45262359 IC50 = 10030 nM T69494 CXA7V0 45262360 IC50 > 10000 nM T69494 C50BJO 45263862 IC50 = 80 nM T69494 CWJ5T9 45263863 IC50 = 2 nM T69494 CJ1X5S 45263913 IC50 = 4.1 nM T69494 C85ZQN 45263934 IC50 = 1.5 nM T69494 CQ4DZ8 45265283 IC50 = 1055 nM T69494 C9CTJ3 45265608 Ki = 834 nM T69494 CNA49J 45272354 IC50 = 28000 nM T69494 CKDA64 49796208 IC50 = 3630.78 nM T69494 CSG9X5 49796212 IC50 = 72443.6 nM T69494 C2DNQ4 49796213 IC50 = 38904.51 nM T69494 CB3UN6 49796486 IC50 = 28840.32 nM T69494 CRQ37Y 49796488 IC50 = 7943.28 nM T69494 C1UC3P 49796489 IC50 = 81283.05 nM T69494 CY9X1C 49796493 IC50 = 16982.44 nM T69494 C15BKS 49796529 IC50 = 5140 nM T69494 C1BT0O 49796530 IC50 = 580 nM T69494 CKEP78 49796531 IC50 = 9070 nM T69494 CUXG85 49796532 IC50 = 5100 nM T69494 C9U6DF 49796534 IC50 = 4340 nM T69494 CAE91G 49796535 IC50 = 8620 nM T69494 C4UW6K 49796538 IC50 = 2430 nM T69494 CN1M0D 49796539 IC50 = 1300 nM T69494 CUF24O 49796541 IC50 = 1190 nM T69494 C4DWG5 49796550 IC50 = 10600 nM T69494 CSPO87 49796552 IC50 = 20600 nM T69494 C5XU2H 49796554 IC50 = 2230 nM T69494 CFR8A4 49796556 IC50 = 4020 nM T69494 C7CNI8 49796559 IC50 = 10830 nM T69494 CMY90L 49796563 IC50 = 2800 nM T69494 C5MUZ4 49796565 IC50 = 3850 nM T69494 CD9X0W 54609066 IC50 = 676082.98 nM T69494 C0RU4W 54676387 IC50 = 290 nM T69494 CY8DN2 54680162 IC50 = 34000 nM T69494 C7HW6P 54680399 IC50 = 660693448 nM T69494 CJ3LG0 54684412 IC50 = 218776162.4 nM T69494 C96LIS 54686710 IC50 = 110 nM T69494 C0Z3WH 54696077 IC50 = 40000 nM T69494 CG1SB7 54696453 IC50 > 100000 nM T69494 CCY18S 54697760 IC50 > 100000 nM T69494 CGW94P 54698129 IC50 = 220 nM T69494 CWRH97 54703399 IC50 = 400 nM T69494 C6K1HR 54704589 IC50 > 100000 nM T69494 C80TQO 54705784 IC50 = 10000000 nM T69494 CS01GD 54708009 IC50 = 61000 nM T69494 C35ILF 54713079 IC50 > 100000 nM T69494 C0J2SM 54730140 IC50 = 10000000 nM T69494 COH35G 54730141 IC50 = 9800 nM T69494 C0TGU6 54730142 IC50 = 23 nM T69494 CWP7S6 54730143 IC50 = 19000 nM T69494 CI7TD9 54730144 IC50 = 31000 nM T69494 C6WJK5 54730145 IC50 = 5400 nM T69494 CCTM78 54730146 IC50 = 20000 nM T69494 CDNH90 54730147 IC50 = 1500 nM T69494 C4RY2J 54730148 IC50 > 100000 nM T69494 CDW9M4 54730149 IC50 = 234422881.5 nM T69494 CV2MW7 54730150 IC50 = 134896288.3 nM T69494 C74URX 54730151 IC50 = 41686938.35 nM T69494 C95JTR 54730152 IC50 = 3000 nM T69494 C6IFX2 54730153 IC50 = 562341325.2 nM T69494 CQP75Y 54730154 IC50 = 2900 nM T69494 CEG0V4 54730155 IC50 = 13000 nM T69494 CCSH03 54730156 IC50 = 3300 nM T69494 C8XP5W 56657647 IC50 = 20 nM T69494 CEUL32 56671494 IC50 = 766 nM T69494 C0GAU6 56671495 IC50 = 56 nM T69494 C84KMT 56674947 IC50 = 11000 nM T69494 CV0ID7 56674948 IC50 = 475 nM T69494 CDI84E 71450922 IC50 > 10000 nM T69494 CI86RN 71584181 IC50 = 42657.95 nM T69494 C74DSX 71584183 IC50 = 43651.58 nM T69494 CDZ57V 71584184 IC50 = 72443.6 nM T69494 C14ALB 71584303 IC50 = 223872.11 nM T69494 CK8FE9 71584304 IC50 = 54954.09 nM T69494 C0LQ6Y 71584305 IC50 = 8511.38 nM T69494 C41APW 71584307 IC50 = 26302.68 nM T69494 CC9OB2 71584309 IC50 = 11481.54 nM T69494 C6KCM7 71584311 IC50 = 109647.82 nM T69494 C10LMZ 71584314 IC50 = 50118.72 nM T69494 CL6S4T 71584442 IC50 = 48977.88 nM T69494 CP45OE 71584446 IC50 = 181970.09 nM T69494 COGD58 71716508 IC50 = 74131.02 nM T69494 CZ70PJ 71716509 IC50 = 25118.86 nM T69494 CRKC24 71716510 IC50 = 22908.68 nM T69494 CQ5D8I 71717118 IC50 = 58884.37 nM T69494 CCTN89 71717740 IC50 = 8709.64 nM T69494 CDYX71 71717741 IC50 = 18197.01 nM T69494 C7T5CL 71717743 IC50 = 63095.73 nM T69494 C5HD9S 71718347 IC50 = 537031.8 nM T69494 CH05NM 71718947 IC50 = 10232.93 nM T69494 CAKP90 71718948 IC50 = 6025.6 nM T69494 C9C1SM 71719559 IC50 = 38018.94 nM T69494 C6U0YD 71719560 IC50 = 70794.58 nM T69494 C7HBZ1 71720158 IC50 = 91201.08 nM T69494 CVIM84 71720799 IC50 = 109647.82 nM T69494 C2F1EX 71720800 IC50 = 229086.77 nM T69494 C8I3MR 71740897 IC50 = 11000 nM T69494 CXJL58 118705656 IC50 = 7762.47 nM T69494 CN63WP 129766223 IC50 = 13400 nM T69494 C8ILY3 135410326 IC50 = 7079457.84 nM T69494 CJZF28 135411159 IC50 = 37 nM T69494 C24CLY 135422276 IC50 = 95499.26 nM T69494 C1WHX8 135429834 IC50 = 1400 nM T69494 CVQ58A 135433790 IC50 = 12 nM T69494 C1P7NC 135439447 IC50 = 33 nM T69494 CAV4R0 135439450 IC50 = 3300 nM T69494 C4YBD2 135460773 IC50 = 910 nM T69494 CF35ZC 135490640 IC50 = 4400 nM T69494 CL8TH4 135522010 IC50 > 100000 nM T69494 CPLD78 135522020 IC50 = 170 nM T69494 C21BFM 135528327 IC50 = 53 nM T69494 C65SAN 135881802 IC50 = 3400 nM T69494 C9C3LB 136056476 IC50 = 2100 nM T69494 CXHY90 136250345 IC50 = 57543.99 nM T69494 CP8HS9 136250348 IC50 = 33113.11 nM T69494 C5IHZ6 136259934 IC50 = 213796.21 nM T69494 C1C2PD 145949977 Ki > 10000 nM T69494 C5Z1LS 145952217 Ki > 10000 nM T69494 CSA16D 145952244 Ki > 10000 nM T69494 CD8I3S 145953412 Ki > 10000 nM T69494 C1AMD5 145955192 Ki > 10000 nM T69494 CGM3L7 145957163 Ki > 10000 nM T69494 C3W0QX 145957790 Ki > 10000 nM T69494 C7GH8Z 145960052 Ki > 10000 nM T69494 CKIQ23 145972645 Ki > 10000 nM T69494 CYNV83 155514509 IC50 = 40000 nM T69494 C8C9SA 155516707 IC50 = 33000 nM T69494 C5QI0C 155532410 IC50 = 11000 nM T69494 CP9TR0 10324985 Ki > 10000 nM T69494 D00ZKW 1228 IC50 = 220 nM T69494 D01LDO 1617430 IC50 = 461 nM T69494 D01SHB 3845 IC50 = 15000 nM T69494 D02WJT 7333 IC50 = 7800 nM T69494 D03RGP 1221 IC50 > 100000 nM T69494 D04DHB 1779 IC50 = 68 nM T69494 D04JJL 14771671 IC50 = 10300 nM T69494 D05KQC 3899541 IC50 = 840 nM T69494 D06NYB 650260 IC50 = 280 nM T69494 D06RFW 13781937 IC50 = 26800 nM T69494 D07QBQ 81143 IC50 = 1800 nM T69494 D08RVB 3035974 IC50 = 107 nM T69494 D0D4IG 10849325 IC50 = 30 nM T69494 D0FT0J 135342 IC50 = 177 nM T69494 D0Q5PC 6468 Ki = 15.3 nM T69494 D0S6HI 2227 IC50 = 9130 nM T69494 D0S6TW 1845 IC50 = 130 nM T40800 D02OZE 2724385 IC50 = 290 nM T40800 CFEQ05 16120562 IC50 = 340 nM T40800 C1K4QJ 16121811 IC50 = 570 nM T40800 CTI1C6 122182551 IC50 = 11000 nM T40800 C1YV8G 122363019 IC50 = 9800 nM T10844 D03HUX 49792852 IC50 > 10000 nM T10844 D0O6WV 24794418 IC50 > 2000 nM T10844 C1XI3D 9929673 IC50 = 100 nM T10844 C0M1ZR 11422615 IC50 = 2900 nM T10844 C9JT4S 11847343 IC50 > 10000 nM T10844 CVZK29 16223008 IC50 > 50000 nM T10844 CY3HW5 46224684 IC50 > 10000 nM T10844 C2Y6QS 50938552 IC50 > 10000 nM T10844 C9NYP4 51036677 IC50 > 10000 nM T10844 C4WRY3 51037112 IC50 > 10000 nM T10844 CRI28Z 51037948 IC50 > 10000 nM T10844 CCN01X 71547862 IC50 > 10000 nM T10844 CY0UC4 90645194 IC50 > 10000 nM T10844 CY7BI2 118706214 IC50 > 10000 nM T10844 D0T8NU 16757525 IC50 > 4000 nM T79332 CEMD65 46863664 IC50 > 10000 nM T79332 D09GVB 10427006 IC50 = 13.4 nM T79332 D0E9UX 25154867 IC50 > 10000 nM T79332 D0NH1E 1383884 IC50 = 5 nM T07448 CIMH03 11852389 Ki = 440 nM T07448 CK16RG 145984220 IC50 = 230 nM T07448 CV8IJ9 145984746 Ki = 6 nM T07448 CWB36A 145984797 Ki = 180 nM T11843 D0E3OF 54678486 IC50 = 8.8 nM T11843 CA6K0Z 54742494 Ki = 44800 nM T11843 C49EQS 54742498 Ki = 74200 nM T11843 CDS19K 54751655 Ki = 79600 nM T11843 CNMV64 70686253 Ki = 68900 nM T11843 CYIN74 155516661 IC50 = 90.2 nM T11843 C4HP0B 155530131 IC50 = 1929 nM T11843 CU56PT 155540911 IC50 = 59 nM T11843 C15VJD 155545987 IC50 = 58.2 nM T11843 CBY58K 155569684 IC50 = 4.5 nM T33931 D03KQF 4011 IC50 = 85000 nM T33931 D0B7NG 2725 IC50 = 42000 nM T33931 CJ9M5X 409443 IC50 > 100000 nM T33931 CUB3O6 646810 IC50 = 75000 nM T33931 C5RFC4 2199015 IC50 = 84000 nM T33931 CFT15I 2199968 IC50 > 100000 nM T33931 CRJ2B0 3447849 IC50 > 100000 nM T33931 CHT0Z2 3668334 IC50 > 100000 nM T33931 CWXM75 3674522 IC50 > 57000 nM T33931 COLH47 4791832 IC50 > 30000 nM T33931 CD5P3W 5542568 IC50 = 5700 nM T33931 CI7MH2 9263860 IC50 = 48000 nM T33931 C64ZSL 43430547 IC50 > 30000 nM T33931 CQ4P5B 44755448 IC50 > 30000 nM T33931 C3NE8O 46931242 IC50 = 2800 nM T33931 CILN45 52936635 IC50 = 28000 nM T33931 C6O8RT 55872720 IC50 = 3700 nM T33931 C2P7SD 56577044 IC50 = 48 nM T33931 CXY3E4 57720618 IC50 = 13000 nM T33931 CY9Z8F 60735522 IC50 > 30000 nM T33931 CB0SA4 61041645 IC50 = 4100 nM T33931 CT9M2C 61041646 IC50 = 6800 nM T33931 C3I5DM 61041804 IC50 = 4100 nM T33931 C84MGB 61242835 IC50 = 6200 nM T33931 C0Y6KO 62947261 IC50 > 30000 nM T33931 C8XEI4 63259457 IC50 > 30000 nM T33931 C0WX5O 70679311 IC50 = 8000 nM T33931 CEW3R6 71598546 IC50 = 62 nM T33931 CUD65X 73333125 IC50 = 450 nM T33931 CHQ18I 73333126 IC50 = 310 nM T33931 C9UDN1 73333127 IC50 = 68 nM T33931 C9K1NV 73333128 IC50 = 39 nM T33931 C4UE6G 73333129 IC50 = 48 nM T33931 CV2SJ4 73333225 IC50 = 53 nM T33931 CF8HO3 73333226 IC50 = 61 nM T33931 CVH9F0 73333227 IC50 = 350 nM T33931 C4PYG2 73333229 IC50 = 160 nM T33931 CBJC52 73333322 IC50 = 130 nM T33931 CRH52C 73333323 IC50 = 1200 nM T33931 CVEN67 73334066 IC50 = 170 nM T33931 CYL3M7 73334067 IC50 = 290 nM T33931 C6T7YX 73334068 IC50 = 350 nM T33931 C70XCT 73334069 IC50 = 120 nM T33931 C8QWP1 73334070 IC50 = 97 nM T33931 CR98DL 73334157 IC50 = 150 nM T33931 CJD9C1 73334158 IC50 = 130 nM T33931 CLRM71 73334159 IC50 = 160 nM T33931 C43NER 73334160 IC50 = 210 nM T33931 CD2HX4 73334161 IC50 = 1100 nM T33931 CC89FN 73334162 IC50 = 1600 nM T33931 COV3R1 73334262 IC50 = 310 nM T33931 CZD0N1 73334263 IC50 = 81 nM T33931 CU3KG0 73334264 IC50 = 120 nM T33931 CMLV27 73334265 IC50 = 740 nM T33931 CD0VK7 73334266 IC50 = 3800 nM T33931 C1SGJ3 73334267 IC50 = 770 nM T33931 C3PYF5 73334361 IC50 = 250 nM T33931 C8H9JF 73334363 IC50 = 74 nM T33931 C8XE1J 73334364 IC50 = 300 nM T33931 CN40ZI 73334365 IC50 = 220 nM T33931 CF9GA5 73334366 IC50 = 340 nM T33931 C69WLM 73334479 IC50 = 3600 nM T33931 CG32QB 73334480 IC50 = 2200 nM T33931 CVE0S2 73334481 IC50 = 620 nM T33931 C2S8XN 73334482 IC50 = 3100 nM T33931 CXJP87 73334483 IC50 = 4500 nM T33931 C57KSE 73334484 IC50 = 110 nM T33931 CAQ18T 73334592 IC50 = 400 nM T33931 CA67YG 73334593 IC50 = 640 nM T33931 CNS84D 73334594 IC50 = 1900 nM T33931 C93HWE 73334595 IC50 = 8000 nM T33931 C87UBE 73334596 IC50 = 110 nM T33931 CKSY83 73334696 IC50 = 88 nM T33931 C36QHM 73334697 IC50 = 220 nM T33931 CF63HU 73334698 IC50 = 130 nM T33931 CQBX27 73334699 IC50 = 210 nM T33931 C0OW1V 73334700 IC50 = 43 nM T33931 C2VFJ9 73349256 IC50 = 3600 nM T33931 CG80NF 73349257 IC50 = 240 nM T33931 COY1J2 73349259 IC50 = 92 nM T33931 CNO9Z5 73350843 IC50 = 280 nM T33931 C8U0ZX 73352326 IC50 = 74 nM T33931 C2OXQ5 76314887 IC50 = 650 nM T33931 C3X7EW 76314888 IC50 = 270 nM T33931 C1YKN5 76314889 IC50 = 360 nM T33931 C4E1BN 76318504 IC50 = 100 nM T33931 CF76CT 76318505 IC50 = 37 nM T33931 CLVA91 76318506 IC50 = 580 nM T33931 C9LNK4 76318507 IC50 = 70 nM T33931 CL87KC 76318508 IC50 = 120 nM T33931 CET23F 76318509 IC50 = 59 nM T33931 C01JLF 76322168 IC50 = 350 nM T33931 C2SEM0 76322169 IC50 = 1300 nM T33931 CRH48X 76322170 IC50 = 320 nM T33931 C5CZV2 76325789 IC50 = 850 nM T33931 CS6GL0 76333019 IC50 = 48 nM T33931 C7IUX5 76333020 IC50 = 1000 nM T33931 CZC8W2 76336632 IC50 = 80 nM T33931 CYQ0B9 76336633 IC50 = 120 nM T33931 CK2N0L 76336634 IC50 = 2400 nM T33931 CS4W5I 76336635 IC50 = 2400 nM T33931 CM6H9O 76336636 IC50 = 390 nM T33931 CL8E1A 83748040 IC50 > 30000 nM T33931 CW25YP 90666882 IC50 = 6900 nM T33931 CQI7D0 90666883 IC50 = 6400 nM T33931 C72IZG 90666884 IC50 > 30000 nM T33931 CCDK35 90666885 IC50 = 23800 nM T33931 C2DCW6 90666886 IC50 > 30000 nM T33931 CXN36J 90666887 IC50 = 8700 nM T33931 CG2S0B 90666888 IC50 = 21000 nM T33931 C19VSG 90666889 IC50 = 6700 nM T33931 CBG12J 90666890 IC50 = 13300 nM T33931 C90LPT 90666891 IC50 = 16000 nM T33931 C0IOH4 90666892 IC50 = 2400 nM T33931 D0F5LH 4634 IC50 > 54000 nM T33931 D0W9RR 57339144 IC50 = 24 nM T61746 D00UVA 11556711 IC50 = 11000 nM T61746 D0SH3I 387447 IC50 > 30000 nM T61746 D0V3YT 10324367 IC50 = 6200 nM T61746 D0X9CH 3010818 IC50 = 210 nM T61746 D06KJQ 42601552 IC50 = 26000 nM T61746 D0H2UB 5361 IC50 > 30000 nM T61746 D0J6AU 10152654 IC50 = 1034 nM T61746 D0HM5J 118253852 IC50 > 20000 nM T61746 D0KG9M 19910 Ki = 39500 nM T61746 D00QHT 183798 Ki = 6900 nM T61746 D01LNG 10201696 IC50 = 61 nM T61746 D04ZIJ 5478883 IC50 = 4260 nM T61746 D0G5ZE 72430 Ki = 24 nM T61746 D0T5PH 6918602 Ki = 13 nM T61746 C0RFA2 3102 IC50 = 288800 nM T61746 CU27VZ 12050 IC50 > 100000 nM T61746 CSA74D 13057 Ki = 111000 nM T61746 C05HLN 26030 IC50 = 600 nM T61746 CYNF54 114619 IC50 = 69.7 nM T61746 CK84SO 123664 Ki = 3.36 nM T61746 C1W9IE 131790 IC50 = 2.28 nM T61746 C0S2PU 152128 IC50 = 45.1 nM T61746 C54ITW 155664 IC50 = 9400 nM T61746 CV8A4D 163098 IC50 > 10000 nM T61746 CM3IB1 245295 Ki = 72000 nM T61746 C8OHY9 254021 IC50 > 10000 nM T61746 CHU6D4 343829 Ki = 84000 nM T61746 C07JLH 404672 Ki = 6900 nM T61746 C6J4GA 446403 Ki = 1 nM T61746 C3YF4P 462382 Ki = 12 nM T61746 C5XV2G 481422 IC50 > 1000000 nM T61746 CW1KP3 481437 IC50 > 300000 nM T61746 C9EAL6 482277 IC50 > 75000 nM T61746 C58PLQ 482278 IC50 > 75000 nM T61746 C2G9IH 482279 IC50 > 75000 nM T61746 C5L4ED 482280 IC50 > 75000 nM T61746 CTW1J9 482282 IC50 > 75000 nM T61746 CK0O9U 482283 IC50 > 75000 nM T61746 CX0SQ5 482284 IC50 > 75000 nM T61746 C6Y5SA 482285 IC50 > 75000 nM T61746 C2D7MH 482286 IC50 > 75000 nM T61746 CAZV26 482287 IC50 > 75000 nM T61746 C2QP9I 482288 IC50 > 75000 nM T61746 C3L9TI 482289 IC50 > 75000 nM T61746 CO3N0A 482290 IC50 > 75000 nM T61746 CZ15KR 482291 IC50 > 75000 nM T61746 C0HV7G 482292 IC50 > 75000 nM T61746 CC1RP8 483672 IC50 > 900000 nM T61746 C1MY6Z 490002 Ki = 6.1 nM T61746 CHF5A4 578663 IC50 = 198000 nM T61746 COMJ65 646525 IC50 = 1990 nM T61746 C1K2FB 647599 IC50 = 1260 nM T61746 C5UQF7 651936 IC50 = 1750 nM T61746 CCKZ79 668744 IC50 = 55000 nM T61746 CRY54Z 690107 IC50 > 10000 nM T61746 C0ER8S 767161 IC50 = 10100 nM T61746 CDVJ42 767163 IC50 = 58300 nM T61746 CE10WO 776842 IC50 = 7300 nM T61746 CJ4MR9 782422 Ki = 97000 nM T61746 C65UJT 980235 IC50 = 17660 nM T61746 CQ2R0M 1011274 IC50 = 5200 nM T61746 C2PRY6 1269450 IC50 = 26900 nM T61746 C25SXA 1440071 IC50 = 37140 nM T61746 CO4AB7 2264784 IC50 = 64800 nM T61746 C0PEK1 2829612 Ki = 153000 nM T61746 C6BI2C 2843953 Ki = 127000 nM T61746 CT8KV2 3001308 IC50 > 10000 nM T61746 CTE79D 3011892 Ki = 40000 nM T61746 C08KQP 3032999 IC50 > 10000 nM T61746 CU43OY 3088969 Ki = 3000 nM T61746 CQO0H7 3240114 IC50 = 690 nM T61746 CE70IL 3241895 IC50 = 440 nM T61746 C63ADU 3243128 IC50 = 700 nM T61746 CMW5A9 4430623 Ki = 34000 nM T61746 C2ZN0V 4479093 IC50 = 150000 nM T61746 CR2ND4 5287468 Ki = 500 nM T61746 CW6D7Z 5287498 IC50 = 5200 nM T61746 CB6H0T 5287549 Ki = 100 nM T61746 CESY50 5288259 IC50 > 500 nM T61746 C9E1UW 5288633 Ki = 5200 nM T61746 CN3RY0 5289345 Ki = 1300 nM T61746 CT8I1B 5292405 IC50 = 72300 nM T61746 CO58XD 5311161 IC50 = 300 nM T61746 CLD0C6 5348879 IC50 = 81500 nM T61746 CF1P5H 5430316 IC50 = 22400 nM T61746 CR6B4P 5465605 IC50 > 10000 nM T61746 C8NX4U 5499839 IC50 = 32100 nM T61746 C3B5YE 5728928 IC50 > 100000 nM T61746 C57VBE 5762376 IC50 > 10000 nM T61746 CZ1XU5 5876194 IC50 = 59400 nM T61746 CW94RA 5897251 IC50 > 100000 nM T61746 C3KI5C 5910205 IC50 > 10000 nM T61746 C1DAZ6 6420159 Ki > 100000 nM T61746 CD51MJ 6442675 IC50 = 57680 nM T61746 C1TE7J 6610318 IC50 = 80 nM T61746 C0XQP7 6917747 IC50 > 100000 nM T61746 CG2A7X 7028541 IC50 = 52300 nM T61746 C9G0KZ 7057919 IC50 = 380000 nM T61746 C54FUT 7272330 IC50 = 17.7 nM T61746 C7WP6J 8194707 IC50 > 100000 nM T61746 CUXQ12 8832875 IC50 > 100000 nM T61746 C2GV5W 8854795 IC50 > 100000 nM T61746 CN26IL 9547980 Ki > 30000 nM T61746 CF40ZX 9562299 IC50 > 10000 nM T61746 C3QN6S 9571439 IC50 > 10000 nM T61746 CLE53W 9580655 IC50 > 10000 nM T61746 CC2ZY8 9580662 IC50 > 10000 nM T61746 CT3Y9G 9580665 IC50 > 10000 nM T61746 CE42MQ 9809035 Ki = 700 nM T61746 CB32AH 9812750 IC50 = 2000 nM T61746 CQ1NG7 9815041 IC50 > 10000 nM T61746 CIX3A6 9816412 IC50 = 1400 nM T61746 CLTO67 9821317 IC50 > 10000 nM T61746 COBW38 9821383 IC50 = 2.24 nM T61746 C9F7PL 9825191 Ki > 150000 nM T61746 C0N4DH 9825355 IC50 = 49 nM T61746 C8W9ER 9827472 Ki = 6900 nM T61746 CN51PR 9829299 Ki = 11000 nM T61746 CK7B2P 9829646 IC50 = 1.8 nM T61746 C2AI0Z 9834360 IC50 = 4200 nM T61746 CLND75 9835685 IC50 = 300 nM T61746 COAM65 9844151 Ki = 32 nM T61746 C2VX4Z 9848148 Ki = 28 nM T61746 C8TL5X 9855884 IC50 = 250 nM T61746 C6Z4WX 9868717 Ki = 7300 nM T61746 CL4VY9 9874885 Ki = 44000 nM T61746 CVS7N2 9877581 IC50 = 500 nM T61746 CC3X2P 9877623 IC50 = 500 nM T61746 CS3C0L 9887581 IC50 > 75000 nM T61746 C7M0IP 9888995 IC50 = 150 nM T61746 C8P5LN 9891030 Ki = 18000 nM T61746 C8HI1R 9891108 IC50 = 12.2 nM T61746 CIBS75 9899272 IC50 = 1100 nM T61746 C2JCM5 9902742 IC50 > 10000 nM T61746 C5XS2F 9904539 Ki = 37000 nM T61746 CR1CL8 9906366 Ki = 1790 nM T61746 CALH63 9908450 Ki = 3843 nM T61746 C7CM6Z 9913250 IC50 = 9.4 nM T61746 CJ6M8N 9915812 IC50 > 300000 nM T61746 C78CYD 9920989 IC50 = 75000 nM T61746 CXD2Y6 9926586 IC50 > 10000 nM T61746 CT74FA 9933804 IC50 = 350 nM T61746 CNR6D5 9948720 IC50 = 940 nM T61746 C0PJ2U 9964915 IC50 = 300 nM T61746 C4WFJ2 9980678 Ki = 34700 nM T61746 CF5W3H 9984343 Ki = 4 nM T61746 CIJ5L2 9987080 IC50 = 9500 nM T61746 CLB5G0 10025017 IC50 > 500 nM T61746 CU1EF5 10047111 IC50 = 12200 nM T61746 C68HGW 10047261 IC50 = 123 nM T61746 C2N9CS 10062713 IC50 = 27 nM T61746 C5X2TU 10069167 Ki = 27 nM T61746 C6O8RU 10072812 IC50 = 6010 nM T61746 CP6Y5W 10076044 Ki = 300 nM T61746 CD6L1T 10098422 Ki = 693 nM T61746 CSO9B2 10099774 Ki > 1000 nM T61746 CA5N3E 10111943 IC50 = 26 nM T61746 CFC3Q8 10120133 IC50 = 9800 nM T61746 C6AZ3B 10120903 IC50 = 870000 nM T61746 CGF5W8 10121332 IC50 = 446 nM T61746 C97NJR 10121949 Ki = 23000 nM T61746 CI3WQ9 10122378 IC50 = 935 nM T61746 CENB09 10122445 IC50 = 383 nM T61746 C7XOA0 10127183 IC50 = 7392 nM T61746 CSO96K 10127748 IC50 = 3600 nM T61746 CKZ15P 10129236 IC50 > 5000 nM T61746 CJ79ZX 10138553 IC50 = 379 nM T61746 CLID02 10144235 Ki = 73000 nM T61746 C8O9WX 10144519 IC50 = 360 nM T61746 CVH3A1 10145940 IC50 = 474 nM T61746 C1WOS4 10146227 IC50 = 19 nM T61746 CI4M8T 10146748 IC50 = 158 nM T61746 CQ3YD8 10150891 IC50 = 1155 nM T61746 C8DQG0 10154619 IC50 > 10000 nM T61746 C9VFI4 10161284 IC50 = 2900 nM T61746 C1Q2EX 10164497 Ki = 98 nM T61746 CDX7R4 10164961 IC50 = 31000 nM T61746 C5B1HM 10165557 IC50 = 12000 nM T61746 C09ALX 10165785 Ki = 32 nM T61746 CR62PT 10165786 Ki > 1000 nM T61746 CTJ7R3 10166544 IC50 = 10000 nM T61746 CDRE91 10167323 Ki = 57000 nM T61746 C2RM3E 10167550 IC50 = 1535 nM T61746 CU0BN5 10168098 IC50 = 126 nM T61746 CB6ZH0 10168228 IC50 = 341 nM T61746 CZ1A8U 10173731 IC50 = 1400 nM T61746 C5NEX6 10174161 IC50 > 5000 nM T61746 C1YR4T 10174359 IC50 > 2000 nM T61746 CD4G7F 10179450 IC50 = 93 nM T61746 CTON03 10179451 IC50 = 1812 nM T61746 C07GUT 10184761 Ki = 22000 nM T61746 C4M3SG 10186046 IC50 = 3500000 nM T61746 CCO7A6 10187105 Ki = 10000 nM T61746 CP2M1T 10187189 Ki > 1000 nM T61746 C9WTI5 10187190 Ki > 1000 nM T61746 C0SF7U 10187920 IC50 = 27000 nM T61746 CWMV50 10190314 IC50 = 369 nM T61746 CKZ1A0 10194354 IC50 = 2374 nM T61746 CZD7A6 10194447 IC50 = 4818 nM T61746 CA2UH4 10194634 IC50 = 5939 nM T61746 CO7XD6 10198366 IC50 = 150 nM T61746 C5T8PK 10198752 IC50 = 200 nM T61746 CQ8YM3 10199981 Ki = 2700 nM T61746 CL9DW3 10200425 IC50 = 2405 nM T61746 CS3IP7 10210867 IC50 = 32000 nM T61746 C1WL9J 10211340 Ki = 1100 nM T61746 C4RW7F 10211405 IC50 = 1260 nM T61746 C1F9SP 10216231 IC50 = 5903 nM T61746 C1Y3QZ 10216510 IC50 = 6086 nM T61746 C5GSN6 10216511 IC50 = 2476 nM T61746 CT8K5D 10231379 IC50 = 20 nM T61746 C4OZ5K 10231447 IC50 = 45000 nM T61746 CJBI61 10237771 IC50 = 2993 nM T61746 CFI43Z 10238903 IC50 = 1561 nM T61746 C6A8NV 10252643 Ki = 270 nM T61746 C0ZV3I 10257116 Ki = 6780 nM T61746 C56PLQ 10258908 Ki = 72000 nM T61746 C9SOH2 10271564 IC50 = 554 nM T61746 C1NJF9 10281819 IC50 = 171 nM T61746 C4TNV3 10283187 IC50 = 444 nM T61746 CKX0R7 10287617 IC50 = 3353 nM T61746 CUW38E 10288162 IC50 = 8869 nM T61746 CX23AL 10288163 IC50 > 10000 nM T61746 CY7DQ2 10288811 IC50 > 2000 nM T61746 CV9LB1 10302710 IC50 = 56000 nM T61746 CUQ2R3 10303526 IC50 = 107000 nM T61746 CV5S7B 10303657 IC50 = 870000 nM T61746 CZR02J 10303878 Ki = 2100 nM T61746 C4S2YM 10304728 IC50 = 133 nM T61746 CPT49O 10310362 IC50 = 4699 nM T61746 CO0GQ8 10313520 IC50 = 2300 nM T61746 CMR75W 10318568 IC50 = 300 nM T61746 C78XZT 10341806 IC50 = 60 nM T61746 C7D9XB 10363069 IC50 = 25000 nM T61746 CDY26B 10366413 Ki = 99 nM T61746 CD9ZI0 10373289 Ki = 340 nM T61746 CD45JN 10392931 Ki = 1260 nM T61746 CS7DJ9 10404797 IC50 > 10000 nM T61746 C9IJ6Y 10408700 IC50 = 3600 nM T61746 CDVZ19 10431266 Ki = 4300 nM T61746 CCU90A 10432068 Ki = 70 nM T61746 C8DTH3 10436731 IC50 = 6.8 nM T61746 CS80VR 10438758 Ki = 1100000 nM T61746 CN18SE 10456222 IC50 = 85.1 nM T61746 CXL4O2 10457121 Ki = 3200 nM T61746 C8WK0J 10457697 IC50 = 0.029 ug.mL-1 T61746 C5N9DB 10460031 IC50 > 300000 nM T61746 CK9PX5 10461097 Ki > 1000 nM T61746 C6KJM2 10461790 Ki = 1600 nM T61746 C9M2RV 10483128 Ki > 10000 nM T61746 CW7V0M 10496067 IC50 > 1000 nM T61746 C1MX2S 10499322 Ki = 7800 nM T61746 CQW51O 10506703 IC50 > 300000 nM T61746 CYQB28 10507021 IC50 > 300000 nM T61746 CFNK35 10507077 IC50 = 19000 nM T61746 CHTL13 10507714 Ki > 1000 nM T61746 CZ80TL 10507960 Ki > 1000 nM T61746 CGA7D1 10515827 IC50 = 1500 nM T61746 CZUA37 10531571 Ki > 1000 nM T61746 C7NJQ1 10554839 IC50 > 300000 nM T61746 COP6I9 10566003 IC50 = 780 nM T61746 CR54HQ 10569603 Ki > 10000 nM T61746 C8U1RQ 10593841 Ki > 10000 nM T61746 CN8PB5 10649378 Ki = 45 nM T61746 CM29WH 10663100 IC50 > 1000 nM T61746 CJ7U3O 10668284 IC50 > 10000 nM T61746 C9V5EX 10673009 Ki = 59 nM T61746 CCF8L6 10674356 IC50 = 225000 nM T61746 CRL23A 10674588 Ki > 10000 nM T61746 C9PY4N 10690022 Ki > 10000 nM T61746 C3VCM6 10690823 Ki = 120 nM T61746 CKO6L0 10698950 Ki = 440 nM T61746 CP2WG8 10716501 IC50 > 1000 nM T61746 CDS3M7 10722309 Ki = 46 nM T61746 C0XE7T 10740734 Ki = 45 nM T61746 C7AEI6 10745144 IC50 > 300000 nM T61746 C9SPK8 10770715 IC50 = 1.4 ug.mL-1 T61746 C5SN8Q 10786038 Ki = 23 nM T61746 CD72KH 10788273 Ki = 41 nM T61746 C9AIY1 10793962 Ki = 2600 nM T61746 C9XI7T 10804795 IC50 > 10000 nM T61746 C28DOK 10816650 IC50 > 300000 nM T61746 CGP01V 10817508 IC50 > 300000 nM T61746 CZ4V0F 10832380 Ki > 10000 nM T61746 C78VEK 10837067 Ki > 1000 nM T61746 C1BT8R 10853144 IC50 > 1000 nM T61746 CBK06L 10861643 IC50 = 78 nM T61746 CBWJ85 10862359 IC50 = 2599 nM T61746 CU9A2L 10874453 IC50 = 42 nM T61746 CPAF53 10876251 Ki = 7.29 nM T61746 C1YU4K 10882794 IC50 = 308 nM T61746 CMO9Y1 10886114 Ki = 600 nM T61746 C7YTP5 10887117 Ki = 0.3 nM T61746 C7ZNC2 10892596 IC50 = 34000 nM T61746 CZK49P 10893343 IC50 > 10000 nM T61746 CTZ4G0 10898089 Ki = 1.41 nM T61746 C6WUK7 10898110 Ki = 0.25 nM T61746 CRM1T6 10902697 IC50 = 3000 nM T61746 CWXN58 10902758 Ki > 330 nM T61746 CBJ1I7 10902914 IC50 > 10000 nM T61746 CA30HS 10905508 IC50 = 3433 nM T61746 CA9ZC6 10907387 Ki = 1300 nM T61746 CCOZ95 10907912 IC50 = 5.6 nM T61746 C5X6NA 10924832 IC50 > 10000 nM T61746 C3CH6U 10930003 IC50 = 47 nM T61746 C3VN9H 10931029 Ki = 43 nM T61746 CZG37Y 10938664 IC50 = 5788 nM T61746 CA72YH 10949332 IC50 = 496 nM T61746 CR0P8J 10971179 IC50 > 10000 nM T61746 CK9E8W 10972182 IC50 > 10000 nM T61746 C6ZOI1 10979734 IC50 > 10000 nM T61746 CCFA87 10983274 IC50 = 140 nM T61746 C57TZJ 10985562 Ki = 0.03 nM T61746 CA3NG9 10993428 IC50 = 8055 nM T61746 C4E0HT 11007209 Ki = 0.13 nM T61746 CM9Z5T 11012257 IC50 > 10000 nM T61746 C5XHI0 11014664 IC50 = 1744 nM T61746 CC6OQ2 11017520 Ki = 40 nM T61746 C56FMI 11027472 Ki = 111.8 nM T61746 CL19TE 11028356 Ki = 45.4 nM T61746 CY72BF 11034349 IC50 > 10000 nM T61746 CQXP76 11050104 Ki = 1700 nM T61746 C5C8TK 11061638 Ki = 0.12 nM T61746 CMP6K1 11071803 Ki = 135.9 nM T61746 CY3V4J 11080121 IC50 = 87 nM T61746 C0PSR8 11081485 IC50 > 10000 nM T61746 C1LCH5 11090074 IC50 = 72 nM T61746 CQV98Y 11092936 IC50 = 29 nM T61746 CMC63T 11113842 Ki = 4800 nM T61746 C47YLE 11114029 IC50 = 110 nM T61746 C5O2BF 11132900 IC50 = 31.3 nM T61746 CCA56R 11145060 IC50 < 10 nM T61746 C1FXG8 11145868 IC50 = 10.2 nM T61746 C1WAF8 11145939 IC50 = 2 nM T61746 CN0F8E 11199915 Ki = 18 nM T61746 C2S0QN 11206482 Ki > 330 nM T61746 CFOV37 11237019 IC50 > 1000000 nM T61746 CCH6N4 11283555 IC50 = 7740 nM T61746 C2M7UP 11343089 IC50 > 30000 nM T61746 C5X1VW 11351327 IC50 = 1000 nM T61746 C3X7AL 11432299 IC50 > 1000000 nM T61746 C1AT2Z 11453155 IC50 = 287 nM T61746 CL1D2Z 11471738 IC50 = 520 nM T61746 CZLF20 11494632 Ki > 330 nM T61746 CR2M4H 11494672 Ki > 330 nM T61746 CM41QW 11494775 Ki = 3000 nM T61746 CT8S4U 11496335 Ki = 280 nM T61746 CC92RV 11501571 Ki = 8600 nM T61746 CFI8L5 11502586 IC50 = 1400 nM T61746 CK5JM6 11503223 Ki = 420 nM T61746 CY4A7V 11504785 Ki = 740 nM T61746 CCH09G 11507712 Ki = 110000 nM T61746 CHI9N5 11512144 Ki = 690 nM T61746 CF20TJ 11514361 Ki > 330 nM T61746 C23DKS 11516307 IC50 = 4200 nM T61746 CDA9F5 11517167 Ki = 13000 nM T61746 C6B5UF 11520360 IC50 > 150000 nM T61746 C87YFV 11523212 Ki = 3460 nM T61746 C6D2VI 11525733 Ki = 340 nM T61746 CQ69XF 11533114 Ki = 1700 nM T61746 C2BT3L 11533910 Ki = 840 nM T61746 C98EQF 11545899 IC50 = 270 nM T61746 C6XK8V 11547772 Ki = 890 nM T61746 C65NQY 11550481 Ki > 330 nM T61746 CG57TI 11551229 Ki > 150000 nM T61746 C3BTN5 11556651 IC50 = 29000 nM T61746 CXTQ39 11558838 Ki > 150000 nM T61746 CF9DE7 11561418 Ki = 3100 nM T61746 CA61ZJ 11562424 Ki = 510 nM T61746 CKH13D 11562461 Ki = 640 nM T61746 CTN57Q 11562607 Ki = 76000 nM T61746 CMH1V5 11563622 IC50 = 54000 nM T61746 CB3W8O 11565199 Ki > 15000 nM T61746 CPY84F 11569750 Ki = 380 nM T61746 CW1O0M 11569883 Ki = 540 nM T61746 C8T5DM 11570453 IC50 > 150000 nM T61746 C1TV6S 11580329 Ki = 70000 nM T61746 C9YNX2 11581727 Ki = 5170 nM T61746 CB1L7I 11583999 IC50 = 77000 nM T61746 C73VCU 11584899 Ki = 193 nM T61746 CJG6T3 11585276 Ki = 24 nM T61746 CER65Q 11588182 Ki > 330 nM T61746 CUX70T 11588744 Ki = 9300 nM T61746 C2Y6JE 11590993 Ki = 870 nM T61746 C1A6ME 11592350 IC50 = 40 nM T61746 CLV84W 11594784 Ki = 99000 nM T61746 CR9VG2 11599767 IC50 > 150000 nM T61746 C85WBA 11599792 Ki = 114000 nM T61746 CQZ5T4 11602113 Ki > 330 nM T61746 C1NV2U 11605163 Ki = 740 nM T61746 C98KMP 11612451 Ki = 3800 nM T61746 CZU5E4 11613136 Ki = 910 nM T61746 CW0T9J 11613973 IC50 > 150000 nM T61746 CK0AN9 11616537 Ki = 1100 nM T61746 C7W8JG 11616689 Ki > 330 nM T61746 CE8WO5 11618337 Ki = 680 nM T61746 CTL1P3 11618795 Ki = 1800 nM T61746 CH21OU 11623464 Ki > 330 nM T61746 CQ7KD1 11623853 Ki = 63000 nM T61746 CUS5Q4 11630803 Ki = 10000 nM T61746 C3XO5G 11631355 Ki > 330 nM T61746 C70VTY 11631953 Ki = 7900 nM T61746 CLUA24 11636269 IC50 > 150000 nM T61746 CLMY50 11641509 Ki = 1100 nM T61746 CNH8C7 11646581 Ki = 5350 nM T61746 CILB73 11649751 Ki > 100000 nM T61746 C8NZX4 11651881 Ki > 330 nM T61746 CJRN14 11655672 Ki = 1400 nM T61746 C5ZOM0 11656060 IC50 = 82 nM T61746 CD2F7P 11656780 IC50 = 100 nM T61746 CO76PW 11659287 Ki > 330 nM T61746 C0Q7AH 11662896 Ki = 530 nM T61746 C0D7NS 11663810 Ki = 670 nM T61746 CYR86V 11664755 IC50 = 38000 nM T61746 CSD3H5 11666846 Ki > 330 nM T61746 C5SJ9K 11669355 IC50 > 10000 nM T61746 C13TGX 11671560 Ki = 56000 nM T61746 CT0OZ8 11673881 Ki > 150000 nM T61746 C1BGL5 11677886 Ki = 1300 nM T61746 C23ZVP 11678241 Ki > 1000 nM T61746 C27LJY 11678922 Ki = 150 nM T61746 CDNH37 11680631 Ki > 150000 nM T61746 C1Q2OT 11682028 Ki = 1300 nM T61746 C6Q8KO 11682184 Ki = 3100 nM T61746 CNB67S 11684874 Ki = 760 nM T61746 C38REW 11695166 Ki > 150000 nM T61746 C6F1GI 11695261 Ki > 330 nM T61746 CJB3E9 11695584 Ki = 5200 nM T61746 C0OC5V 11696208 Ki = 8300 nM T61746 C5H2GL 11696621 Ki > 330 nM T61746 CHP6U3 11699298 Ki = 1400 nM T61746 C5UEI7 11703527 IC50 = 2340 nM T61746 C9X6PV 11703830 Ki = 2100 nM T61746 CU57OC 11705307 IC50 = 65.6 nM T61746 C0Y5XV 11705688 Ki = 1500 nM T61746 CRZ6T0 11709547 Ki > 330 nM T61746 CT4QY5 11710096 Ki > 330 nM T61746 C5FZ1J 11710873 IC50 = 2512 nM T61746 C5ME9N 11716536 Ki > 330 nM T61746 C26RZY 11717535 Ki = 2300 nM T61746 CRSM12 11730723 IC50 = 16.9 nM T61746 CF3LI6 11731499 IC50 = 30.7 nM T61746 CDS4P0 11743922 Ki = 1950 nM T61746 CY63BP 11761693 IC50 = 40 nM T61746 C9WY8H 11763098 IC50 > 1000 nM T61746 C8EZR3 11763189 Ki = 45 nM T61746 CGU6I7 11767007 Ki = 42.7 nM T61746 CD73UO 11768265 Ki = 13 nM T61746 C8D7BS 11771234 Ki > 10 nM T61746 CYRC95 11800689 IC50 = 59000 nM T61746 CDJH89 11811557 IC50 = 3843 nM T61746 CZ1YB3 11824245 IC50 > 10000 nM T61746 C6QOP0 11824460 IC50 = 591 nM T61746 C1M9PK 11827945 IC50 = 18 nM T61746 C7KS4F 11849205 Ki = 6990 nM T61746 CDS3P8 11849206 Ki = 4420 nM T61746 CK8QP3 11849207 Ki = 340 nM T61746 CAX2I8 11849208 Ki = 110 nM T61746 CP21OF 11849209 Ki = 2590 nM T61746 C12XMU 11849702 Ki = 1480 nM T61746 C4LAJ0 11849703 Ki = 2540 nM T61746 C5O8YF 11849704 Ki = 1480 nM T61746 CX1A2R 11849705 Ki = 4610 nM T61746 CN02JP 11849751 Ki = 3750 nM T61746 C3W1SA 11849752 Ki = 5400 nM T61746 CM69HK 11849753 Ki = 4180 nM T61746 C6HG9B 11849754 Ki = 230 nM T61746 CA2BX6 11849755 Ki = 90 nM T61746 C13ZOW 11849756 Ki = 6900 nM T61746 COA94E 11849757 Ki = 12100 nM T61746 C0YB2W 11849844 Ki = 3500 nM T61746 CERY85 11849845 Ki = 2470 nM T61746 CH75EO 11849846 Ki = 5450 nM T61746 CRXO59 11857300 IC50 = 337 nM T61746 CDOG76 11857302 IC50 > 10000 nM T61746 C3QN1E 11983275 Ki = 220 nM T61746 C7FV2Q 12404626 Ki = 176000 nM T61746 CP4H9E 12737307 Ki = 77000 nM T61746 CHW30V 12967046 IC50 = 1.3 ug.mL-1 T61746 C53JDX 12968472 IC50 = 138 nM T61746 C31MCN 13186896 IC50 > 100000 nM T61746 CA78NJ 13386706 Ki = 4341000 nM T61746 C2KW1D 13814218 IC50 = 232000 nM T61746 C4JQR9 14060550 Ki > 330 nM T61746 C9WC6M 14655218 Ki > 330 nM T61746 C3OI2T 15017709 IC50 = 97.7 nM T61746 CM7H4S 15283376 Ki > 330 nM T61746 CT48FA 15407997 IC50 > 300000 nM T61746 CN91PY 15547226 IC50 > 50000 nM T61746 CCGS52 15547237 IC50 = 1300 nM T61746 CI8QZ5 15567852 Ki > 330 nM T61746 CVO9K6 15858812 IC50 = 1760 nM T61746 C6FCZ8 15949750 Ki = 33300 nM T61746 C2QO1B 15955412 Ki = 3900 nM T61746 CHC31Q 15985697 IC50 = 3453 nM T61746 C9LW6H 15985754 IC50 = 953 nM T61746 CQ5F9T 16045426 IC50 = 987 nM T61746 CY0FX8 16061496 IC50 > 10000 nM T61746 C08XJK 16090559 Ki > 10000 nM T61746 CTIV96 16090560 Ki > 10000 nM T61746 C2QWA9 16090561 Ki > 10000 nM T61746 CJBT92 16090562 Ki > 10000 nM T61746 CU6KB8 16090563 Ki > 15000 nM T61746 C6D4FQ 16655063 IC50 = 13 nM T61746 C5FUL9 16661369 IC50 > 100000 nM T61746 CUTI57 16661526 IC50 > 100000 nM T61746 C26JIW 16661682 IC50 > 100000 nM T61746 C6XPN4 16664855 IC50 = 1 nM T61746 C8XLP2 16720100 Ki > 15000 nM T61746 C4P8ZV 16720327 Ki > 15000 nM T61746 CUA19Y 16760339 Ki = 2400 nM T61746 CYA5V6 16760340 Ki = 750 nM T61746 CKA87T 17945762 IC50 = 1903 nM T61746 C7WD4Z 18628647 IC50 = 3329 nM T61746 CR7B9L 18628679 IC50 > 10000 nM T61746 CHA0S3 18628693 IC50 = 1075 nM T61746 CU3NM9 18628717 IC50 > 10000 nM T61746 C71IFZ 18628739 IC50 = 6369 nM T61746 CUSD12 18628799 IC50 = 3343 nM T61746 C5ZRU1 19540655 IC50 > 100000 nM T61746 CLM2E4 19959068 IC50 = 32000 nM T61746 C8O5CM 20828112 Ki = 349000 nM T61746 C34QUK 21309371 IC50 > 50000 nM T61746 C2KBL6 22972497 IC50 > 10000 nM T61746 CD5R3V 22972573 IC50 = 2227 nM T61746 CFY7O6 22988664 Ki = 32000 nM T61746 C6YW0C 23240737 Ki = 1300 nM T61746 C15TFI 23240738 Ki = 6000 nM T61746 C2NRA7 23240739 Ki = 9300 nM T61746 CKW6Q8 23626706 IC50 = 1104 nM T61746 CZ8DI1 23643986 Ki = 1100 nM T61746 CZPF48 23648277 IC50 = 280 nM T61746 CHU59C 23648278 IC50 = 417 nM T61746 CA74XT 23648279 IC50 = 8029 nM T61746 C2I6RW 23648280 IC50 = 170 nM T61746 CCJ8M5 23648281 IC50 = 9724 nM T61746 C9C0HK 23648282 IC50 = 3854 nM T61746 CC50JD 23648283 IC50 = 1980 nM T61746 CS1VW7 23648284 IC50 = 2777 nM T61746 CUQH43 23648285 IC50 = 1844 nM T61746 CM52JD 23648286 IC50 = 1319 nM T61746 CE09VM 23648287 IC50 = 4041 nM T61746 C1FRI4 23648288 IC50 > 10000 nM T61746 C9RNB7 23648289 IC50 = 7280 nM T61746 C4J5MD 23648290 IC50 = 3453 nM T61746 CY20DH 23648291 IC50 = 6629 nM T61746 CF7O3H 23648292 IC50 = 3612 nM T61746 CKI1W5 23648293 IC50 = 2971 nM T61746 CN5S3K 23648294 IC50 = 8507 nM T61746 CTB69E 23648295 IC50 = 4813 nM T61746 C31XJH 23648296 IC50 = 1360 nM T61746 C5ECI8 23648297 IC50 > 10000 nM T61746 CB7T3I 23648298 IC50 > 10000 nM T61746 CVF2M6 23648299 IC50 > 10000 nM T61746 CRZ56K 23648300 IC50 = 1605 nM T61746 CQ1C8H 23648301 IC50 = 1337 nM T61746 CQFD10 23648302 IC50 = 1660 nM T61746 CFR23Q 23648303 IC50 = 6984 nM T61746 C0FBS2 23648304 IC50 > 10000 nM T61746 C67AYX 23648305 IC50 > 10000 nM T61746 CN6R9M 23648306 IC50 = 4073 nM T61746 C85PXH 23648308 IC50 = 1873 nM T61746 CVH82R 23648309 IC50 = 483 nM T61746 COZK65 23648310 Ki > 30000 nM T61746 C6P3YR 23648430 IC50 = 310 nM T61746 C5AQX8 23648431 IC50 = 170 nM T61746 C0M8FS 23648434 IC50 = 130 nM T61746 CD7R1S 23648435 IC50 = 72 nM T61746 CF9H8N 23648436 IC50 = 79 nM T61746 CZG5U1 23648437 IC50 = 71 nM T61746 CF68MH 23648438 IC50 = 40 nM T61746 C2C5YA 23648440 IC50 = 68 nM T61746 C7DBS2 23648441 Ki > 1000 nM T61746 C1YTO9 23648449 IC50 > 10000 nM T61746 CJO2P4 24776563 IC50 > 30000 nM T61746 CR8L2N 24776564 IC50 > 30000 nM T61746 C3U0QR 24776565 IC50 > 30000 nM T61746 CV9F0D 24776566 IC50 > 30000 nM T61746 COZ5C9 24776567 IC50 > 30000 nM T61746 C28RDA 24776568 IC50 > 30000 nM T61746 C9KHL2 24776569 IC50 > 30000 nM T61746 CA4KQ3 24776683 IC50 > 30000 nM T61746 C92NZG 24776926 IC50 = 19050 nM T61746 CN1R6S 24776927 IC50 = 17700 nM T61746 CT06JY 24776928 IC50 > 30000 nM T61746 CHF5Y7 24776929 IC50 > 30000 nM T61746 CO3W9N 24776931 IC50 > 30000 nM T61746 C2Y8JF 24776932 IC50 > 30000 nM T61746 CPBT05 24777048 IC50 > 30000 nM T61746 CM4KX2 24777049 IC50 > 30000 nM T61746 C6ACK9 24777050 IC50 > 30000 nM T61746 CCP4V6 24777300 IC50 > 30000 nM T61746 C8JR9Q 24777301 IC50 > 30000 nM T61746 CYMF31 24777302 IC50 > 30000 nM T61746 CA04CB 24777303 IC50 = 5430 nM T61746 CJ3N1A 24777429 IC50 > 30000 nM T61746 CBI96T 24777430 IC50 > 30000 nM T61746 CAF5Y4 24777431 IC50 > 30000 nM T61746 CB96XZ 24778049 IC50 = 23600 nM T61746 CK74OH 24778050 IC50 > 30000 nM T61746 CQHR89 24778051 IC50 > 30000 nM T61746 CUG91O 24778054 IC50 > 30000 nM T61746 CF30JZ 24778183 IC50 > 30000 nM T61746 CB50GN 24778184 IC50 > 30000 nM T61746 CUP2D4 24778185 IC50 > 30000 nM T61746 C15VPF 24778187 IC50 > 30000 nM T61746 CFWK93 24778188 IC50 > 30000 nM T61746 CF9WJ1 24778189 IC50 > 30000 nM T61746 CVS50O 24778317 IC50 > 30000 nM T61746 CC4TG6 24778318 IC50 > 30000 nM T61746 CTV8S9 24778319 IC50 > 30000 nM T61746 CYP8K1 24778320 IC50 > 30000 nM T61746 CPT6I2 24778321 IC50 > 30000 nM T61746 CKP1F7 24778322 IC50 > 30000 nM T61746 CB64RJ 24778323 IC50 > 30000 nM T61746 C7U5ZK 24778439 IC50 > 30000 nM T61746 CEP4D9 24778440 IC50 = 7690 nM T61746 CH8YB7 24778441 IC50 > 30000 nM T61746 CYCD75 24778442 IC50 > 30000 nM T61746 CB3K0R 24778443 IC50 > 30000 nM T61746 CQ80SX 24778444 IC50 = 1040 nM T61746 CV5P1B 24778445 IC50 > 30000 nM T61746 CGTM78 24800873 Ki = 14500 nM T61746 C1LOF2 24800874 Ki = 3300 nM T61746 CMI4L3 24800875 Ki = 4600 nM T61746 CAXQ09 24801230 Ki = 4400 nM T61746 CT1A2Z 24801231 Ki = 3100 nM T61746 C2O4WK 24801410 Ki = 11000 nM T61746 C5NI0K 24801411 Ki = 4300 nM T61746 CN0VA7 24822701 IC50 > 50000 nM T61746 C2GQ6X 24897809 Ki = 0.43 nM T61746 CJ6G9K 24898026 Ki > 330 nM T61746 CZ21HD 24898027 Ki = 0.68 nM T61746 C3TM0A 24898029 Ki > 330 nM T61746 CQU38W 24900755 IC50 = 46 nM T61746 C2S8VB 24901099 IC50 = 5 nM T61746 CIN28B 24901100 IC50 = 2 nM T61746 CD2EH0 24901101 IC50 = 8 nM T61746 CS7B3F 24901102 IC50 = 158 nM T61746 C0JX5G 24939081 IC50 = 1.4 ug.mL-1 T61746 CGI0U2 25023791 IC50 > 30000 nM T61746 C43JRI 25066441 IC50 = 300 nM T61746 CF54QZ 25129041 IC50 = 3981.07 nM T61746 CDO26T 25129042 IC50 = 1584.89 nM T61746 C57LJM 25129043 IC50 = 1140 nM T61746 C3AT6W 25130088 IC50 = 766 nM T61746 C1FWI6 25133836 IC50 = 2400 nM T61746 CYV1J6 25133837 IC50 = 40000 nM T61746 CBZK08 25133838 IC50 = 1995.26 nM T61746 CP8U3Q 25142042 IC50 = 3520 nM T61746 CC92AI 25142043 IC50 > 2900 nM T61746 C8IFW0 25142172 IC50 > 2900 nM T61746 CD2A6W 25142173 IC50 > 2900 nM T61746 C53OMA 25142175 IC50 > 2900 nM T61746 C7CFR2 25142176 IC50 > 2900 nM T61746 C78RJG 25142177 IC50 > 2900 nM T61746 CS6R4T 25142308 IC50 > 2900 nM T61746 CM2PI4 25142309 IC50 > 2900 nM T61746 CM6FL3 25142310 IC50 > 2900 nM T61746 CWV4F5 25142312 IC50 > 2900 nM T61746 CH52AJ 25142313 IC50 > 2900 nM T61746 COG9V7 25142440 IC50 > 2900 nM T61746 CYL56K 25142444 IC50 > 2900 nM T61746 C3IT4O 25142445 IC50 > 2900 nM T61746 CK7D0V 25142571 IC50 > 2900 nM T61746 CW9KR5 25142573 IC50 > 2900 nM T61746 CZ0G2I 25142574 IC50 > 2900 nM T61746 CNH31I 25142699 IC50 > 2900 nM T61746 CQ9PD6 25142700 IC50 > 2900 nM T61746 CV08DB 25142970 IC50 > 2900 nM T61746 C3C8YJ 25174148 IC50 > 25118.86 nM T61746 C5M1BT 25195691 IC50 > 25118.86 nM T61746 CC7TV3 25204336 IC50 > 10000 nM T61746 C73KLE 25209862 IC50 = 1700 nM T61746 CPCS30 25211573 Ki = 880 nM T61746 C9FWJ4 25219913 IC50 = 76470 nM T61746 CJ04ZN 25234563 IC50 > 10000 nM T61746 CW9JM2 25256832 IC50 > 10000 nM T61746 C3GC7P 25256833 IC50 = 6100 nM T61746 CXU0P9 26794600 Ki = 7096000 nM T61746 C9P0TZ 31538102 Ki = 137000 nM T61746 CEM46K 31538150 Ki = 38000 nM T61746 CTME03 38864605 IC50 = 1810 nM T61746 C26LPI 38864607 IC50 = 28950 nM T61746 CN80BC 38864634 IC50 = 54290 nM T61746 CL96WQ 42633150 IC50 = 231 nM T61746 CZ5F4C 42633340 IC50 = 260 nM T61746 C5XV0H 42633341 IC50 = 9 nM T61746 CZS24P 42633520 IC50 = 41 nM T61746 CI78XT 42633521 IC50 = 87 nM T61746 CU6PL7 42633691 IC50 = 48 nM T61746 CQ9TR8 42633692 IC50 = 122 nM T61746 C6FJW2 42634249 IC50 = 64 nM T61746 C9EN0G 42634411 IC50 = 27 nM T61746 C2ZXJ7 42634578 IC50 = 433 nM T61746 CI25RJ 42634754 IC50 = 54 nM T61746 CZ6B1F 42635119 IC50 = 143 nM T61746 C5X4WG 42635483 IC50 = 79 nM T61746 CZM36T 42641892 IC50 > 10000 nM T61746 CRYH80 42642459 IC50 > 10000 nM T61746 CBD6W5 43414832 Ki = 47000 nM T61746 C25ELB 44143088 IC50 = 10715.19 nM T61746 CYKN50 44156293 Ki = 800 nM T61746 CNM6X8 44218399 IC50 = 53 nM T61746 C8Y9NQ 44219712 IC50 = 3890 nM T61746 CJA68L 44224113 IC50 = 5011.87 nM T61746 C2V5ZT 44224114 IC50 > 10000 nM T61746 C0U9VJ 44224115 IC50 > 10000 nM T61746 C0MZ9D 44224116 IC50 > 10000 nM T61746 CEJ82A 44224117 IC50 = 2511.89 nM T61746 C0KL7D 44224118 IC50 = 5011.87 nM T61746 CE9S0M 44224119 IC50 > 10000 nM T61746 CV1W0Z 44224120 IC50 = 3981.07 nM T61746 C5LDK7 44224121 IC50 = 5011.87 nM T61746 C8UF5Q 44224122 IC50 > 10000 nM T61746 C9YHC5 44224123 IC50 = 7943.28 nM T61746 CA26RI 44224124 IC50 = 10000 nM T61746 CU0PI2 44224125 IC50 > 10000 nM T61746 CRL79W 44224126 IC50 > 10000 nM T61746 C3T0QO 44224127 IC50 > 10000 nM T61746 C81EVM 44224128 IC50 > 10000 nM T61746 C7IY8P 44224129 IC50 > 10000 nM T61746 CYG02V 44224130 IC50 > 10000 nM T61746 CJS1B9 44224131 IC50 = 10000 nM T61746 CN5O8S 44224132 IC50 = 1995.26 nM T61746 C2Q3RP 44224133 IC50 = 7943.28 nM T61746 CZX62T 44224134 IC50 = 5011.87 nM T61746 CP3YA9 44224135 IC50 = 6309.57 nM T61746 CSZH31 44224136 IC50 = 3981.07 nM T61746 CF26LQ 44254142 Ki = 1400 nM T61746 CNS8G1 44254314 Ki = 12400 nM T61746 CVY05S 44254499 Ki = 22900 nM T61746 CAZ9V1 44254582 Ki = 22200 nM T61746 CZ56BP 44263398 IC50 > 20000 nM T61746 C5LJS7 44279083 Ki = 440 nM T61746 C2V7RL 44279437 Ki > 1000 nM T61746 C8D6VK 44282051 IC50 > 75000 nM T61746 C5FY9H 44284219 IC50 = 85.1 nM T61746 CT4FH7 44284304 IC50 = 836 nM T61746 C2ZHC1 44295739 IC50 > 10000 nM T61746 CG3OM8 44304535 Ki = 140000 nM T61746 C0FKB3 44304563 Ki = 7700 nM T61746 CC04TQ 44304591 Ki = 120000 nM T61746 C76OIY 44304610 Ki = 1600 nM T61746 CK8JW5 44304611 Ki = 65000 nM T61746 CZ87NW 44304634 Ki = 52000 nM T61746 COR96D 44304861 Ki > 150000 nM T61746 CXDI94 44317334 Ki = 62 nM T61746 CNBR62 44317343 Ki = 83 nM T61746 CV23BP 44317348 Ki = 99 nM T61746 CT2R6Y 44318099 Ki = 5050 nM T61746 C9O1VP 44319528 Ki = 4 nM T61746 CH9E6N 44321598 Ki = 5 nM T61746 C6EYQ8 44321883 Ki = 52 nM T61746 CTW41Y 44321884 Ki = 3.7 nM T61746 CU7J2P 44321946 Ki = 1.6 nM T61746 C8DX6O 44322591 IC50 = 883 nM T61746 CV2C4T 44322992 IC50 = 3000 nM T61746 CP2IG8 44323050 IC50 = 38 nM T61746 C3KU0G 44323051 IC50 = 1400 nM T61746 C5OT0F 44323240 Ki = 44 nM T61746 C0MF5A 44329571 Ki = 519000 nM T61746 CKB02C 44329582 Ki = 119000 nM T61746 CTN34G 44329585 Ki = 1250 nM T61746 CR1J6F 44329593 Ki = 32200 nM T61746 C3EHF1 44329596 Ki = 1440 nM T61746 C97WPV 44329608 Ki = 1140 nM T61746 CY5KH4 44329643 Ki > 150000 nM T61746 C94FID 44330054 IC50 = 4500 nM T61746 C5CSJ7 44330064 IC50 = 60 nM T61746 CJ5W0G 44332538 Ki = 12920 nM T61746 C1KD2V 44332539 Ki > 10000 nM T61746 C7XQY2 44332540 Ki = 6170 nM T61746 C2FHG7 44332555 Ki = 13220 nM T61746 C6QOU0 44332714 Ki = 10510 nM T61746 C83QDU 44332915 Ki = 4550 nM T61746 C8C4MB 44342381 IC50 > 10000 nM T61746 C7MWQ8 44342499 IC50 = 1000 nM T61746 CQ61OB 44342501 IC50 > 50000 nM T61746 CIBF96 44342511 IC50 = 430 nM T61746 CVK4H3 44342519 IC50 = 390 nM T61746 CN7BH9 44342744 IC50 > 50000 nM T61746 CP2OM5 44342745 IC50 = 430 nM T61746 CMQ6Y0 44342776 IC50 = 30000 nM T61746 C8UKO5 44342803 IC50 > 50000 nM T61746 C6PLY0 44342983 IC50 = 16400 nM T61746 C1IJW5 44343023 IC50 = 12000 nM T61746 C71JRX 44343028 IC50 = 72 nM T61746 COEK09 44343037 IC50 = 400 nM T61746 C61UIS 44343092 IC50 = 2200 nM T61746 CB64RL 44343105 IC50 = 3400 nM T61746 CN5GQ3 44343531 Ki = 3000 nM T61746 CGN37W 44343594 Ki = 200 nM T61746 C47KQO 44343612 Ki = 2000 nM T61746 CW2Z7I 44343748 Ki = 4600 nM T61746 C0TAX2 44345292 Ki > 1000 nM T61746 CD9P4K 44345387 Ki > 1000 nM T61746 C8HP5M 44347822 IC50 = 550 nM T61746 CK0B9C 44347827 IC50 > 10000 nM T61746 CO82ZV 44347993 IC50 > 10000 nM T61746 CLCP51 44348116 IC50 > 10000 nM T61746 CFBI42 44348134 IC50 > 10000 nM T61746 CYEI89 44348185 IC50 = 1249 nM T61746 CV6U1K 44353527 Ki = 4200 nM T61746 CN6B8M 44353535 Ki = 2100 nM T61746 CP5NY3 44353544 Ki = 1200 nM T61746 C5FXE6 44353552 Ki = 9900 nM T61746 CJ0Y3M 44353556 Ki = 2500 nM T61746 C1QG3Z 44353580 Ki = 440 nM T61746 C6T3DA 44353581 Ki = 310 nM T61746 CV6U5Q 44353582 Ki = 630 nM T61746 CMTJ91 44353589 Ki = 350 nM T61746 CM3R5T 44353590 Ki = 2000 nM T61746 CZ2YG8 44353593 Ki = 200 nM T61746 CY6CK7 44353594 Ki = 1200 nM T61746 C6MV2C 44353604 Ki = 13000 nM T61746 CEJ3D8 44353608 Ki = 6400 nM T61746 C0WIP1 44353630 Ki = 2200 nM T61746 C6BQS9 44353632 Ki = 2300 nM T61746 C7DRX0 44353633 Ki = 2800 nM T61746 CS9VG4 44353649 Ki = 4500 nM T61746 C1V8RS 44353769 Ki = 3000 nM T61746 C53QGD 44353782 Ki = 4500 nM T61746 C91OHB 44353783 Ki = 6000 nM T61746 CUY2N7 44353792 Ki = 800 nM T61746 C5XVK9 44353793 Ki = 1800 nM T61746 CH80QO 44353801 Ki = 890 nM T61746 CPA90D 44353812 Ki = 300 nM T61746 CB7P0H 44353839 Ki = 3800 nM T61746 CZ89JO 44353846 Ki = 280 nM T61746 CP3VT2 44353858 Ki = 2000 nM T61746 C5H9VR 44353859 Ki = 340 nM T61746 CNZ2I9 44353889 IC50 = 5 nM T61746 CR6TJ7 44353910 IC50 = 13.3 nM T61746 C9EOS5 44353924 IC50 = 4.9 nM T61746 C4LI8M 44353927 IC50 = 6.5 nM T61746 C6Y7AT 44353935 IC50 = 16.5 nM T61746 C2V6TO 44353936 IC50 > 1000 nM T61746 CG1JP8 44353951 IC50 = 4.1 nM T61746 CX1IL0 44353974 IC50 = 194 nM T61746 CQ1F6V 44353976 IC50 = 5.3 nM T61746 CJA79K 44353977 IC50 = 9.3 nM T61746 C3GV4U 44353978 IC50 = 8.7 nM T61746 C67ZFU 44353986 IC50 = 282 nM T61746 CCJ12M 44354014 IC50 = 5.3 nM T61746 CT7JK8 44354015 IC50 = 8.6 nM T61746 C49VSE 44354016 IC50 = 832 nM T61746 CN85XQ 44354163 IC50 > 300000 nM T61746 CAC2Q0 44356377 IC50 = 1300 nM T61746 CU6KO2 44356379 IC50 > 1000 nM T61746 C6JTS1 44356381 IC50 = 65 nM T61746 CYK6F4 44356399 IC50 = 1400 nM T61746 CUJK15 44356612 IC50 = 120 nM T61746 CBPJ08 44356625 IC50 = 3200 nM T61746 C0DE5P 44356626 IC50 = 100 nM T61746 CI9OQ6 44356637 IC50 = 480 nM T61746 CRA87Z 44356780 IC50 = 3900 nM T61746 CH9L1E 44356846 IC50 = 530 nM T61746 CKS7I4 44357044 IC50 = 30 nM T61746 C35ROP 44357071 IC50 > 1000 nM T61746 CFMJ42 44359521 IC50 = 1900 nM T61746 CR2IZ3 44359576 IC50 = 130 nM T61746 CZ2YK0 44359596 IC50 = 136 nM T61746 CL35EI 44359631 IC50 > 1000 nM T61746 CSG8W5 44359640 IC50 = 652 nM T61746 C9DN5F 44359657 IC50 = 358 nM T61746 CS0AF4 44359658 IC50 = 11.9 nM T61746 C2NVU0 44359684 IC50 = 121 nM T61746 CD10PV 44378627 Ki = 2750 nM T61746 C8SEB4 44378629 Ki = 12100 nM T61746 CAXL14 44378897 Ki = 5260 nM T61746 CA9LC3 44382185 Ki = 9664 nM T61746 C5NH3W 44382186 Ki = 106 nM T61746 CZU70X 44382187 Ki = 167 nM T61746 C3M5CT 44382237 Ki = 12 nM T61746 C3W7CI 44382238 Ki = 7 nM T61746 CUEX04 44382949 Ki > 10000 nM T61746 C9UQN0 44383254 Ki > 10000 nM T61746 CU4CB8 44383255 Ki = 2094 nM T61746 C83ART 44383306 Ki = 658 nM T61746 CP7KW2 44391459 IC50 = 310 nM T61746 C9W3HN 44391474 IC50 = 2.4 nM T61746 CV71WQ 44391475 IC50 = 680 nM T61746 CIG5R6 44393795 IC50 = 158 nM T61746 C78QJO 44394249 Ki = 13000 nM T61746 CQRB69 44394250 Ki = 283000 nM T61746 CTRP74 44394287 IC50 = 5000 nM T61746 CP7X6J 44394353 IC50 > 5000 nM T61746 C79NFU 44394458 IC50 > 12000 nM T61746 C2J6MW 44397423 IC50 = 6200 nM T61746 CRSF50 44397609 IC50 = 60000 nM T61746 CHWX97 44397693 IC50 = 18000 nM T61746 CD73QR 44398649 Ki = 1.3 nM T61746 CHQF16 44398651 Ki = 0.077 nM T61746 C4ALQ9 44398659 Ki = 2600 nM T61746 CGQ20I 44398741 Ki = 0.25 nM T61746 CD18YP 44402055 IC50 > 2000 nM T61746 CU8TB9 44402056 IC50 > 5000 nM T61746 CD4TP7 44402158 IC50 > 13000 nM T61746 CO6BG2 44402160 IC50 = 12000 nM T61746 C0AJC4 44402175 IC50 > 13000 nM T61746 CX9O2Q 44402263 IC50 > 13000 nM T61746 C89MOT 44402291 IC50 > 13000 nM T61746 CFL9B8 44402952 IC50 > 10000 nM T61746 CRZT97 44403028 IC50 > 10000 nM T61746 CY5NW9 44405210 Ki = 590 nM T61746 CP8L2A 44405213 Ki = 3000 nM T61746 CA59MJ 44405279 Ki > 150000 nM T61746 C5GS4Y 44405280 Ki > 150000 nM T61746 CXPM85 44405281 IC50 = 650 nM T61746 CDP93F 44405305 Ki > 150000 nM T61746 CM6Q0Z 44405329 IC50 = 120 nM T61746 C4ZMP9 44408016 IC50 = 32000 nM T61746 C25RIN 44408049 IC50 = 18 nM T61746 C20RAT 44409659 Ki = 120 nM T61746 CA63VX 44409753 Ki = 20 nM T61746 CZ6AD5 44410025 Ki = 22100 nM T61746 C21GXN 44410779 Ki = 18000 nM T61746 CY4H2I 44411981 Ki = 75 nM T61746 CNU4T9 44412155 Ki = 2 nM T61746 CYF1B9 44412339 Ki > 150000 nM T61746 C1J6OW 44412340 Ki > 150000 nM T61746 CU49OM 44412341 Ki = 120000 nM T61746 CDK32G 44412349 Ki = 430 nM T61746 CL82XD 44412354 Ki = 25000 nM T61746 C23ZVR 44412355 Ki = 34000 nM T61746 CV26BC 44412365 Ki = 16000 nM T61746 CX93NW 44412366 Ki = 48000 nM T61746 CZN9T0 44412387 Ki = 93 nM T61746 CY90QW 44412402 Ki = 270 nM T61746 C1HW8F 44412424 Ki = 950 nM T61746 CYDJ14 44412436 Ki = 730 nM T61746 CV49GB 44412437 Ki = 110000 nM T61746 CZ5VW2 44412440 Ki = 7300 nM T61746 CZR1O3 44412502 Ki > 150000 nM T61746 C7VEA8 44414966 Ki = 12100 nM T61746 C9SU1L 44414975 Ki = 119 nM T61746 CA23SL 44414977 Ki = 12000 nM T61746 C0XB2M 44414978 Ki = 37000 nM T61746 CAG5F3 44414992 Ki = 51000 nM T61746 C8JL9C 44415006 Ki = 51000 nM T61746 C0THI1 44415189 IC50 = 88900 nM T61746 CGDY32 44415219 IC50 = 63100 nM T61746 CS6X7V 44426055 IC50 = 519 nM T61746 C8IB2W 44426056 IC50 > 100000 nM T61746 CJ94BD 44430088 IC50 = 495 nM T61746 C61ERA 44430089 IC50 = 396 nM T61746 CU62AV 44430090 IC50 = 320 nM T61746 CRHO67 44430091 IC50 = 316 nM T61746 C27HKY 44430092 IC50 = 271 nM T61746 C4RQ8C 44430093 IC50 = 404 nM T61746 C2DI8G 44430095 IC50 = 150 nM T61746 CV2IX0 44430096 IC50 = 186 nM T61746 CJDT19 44430097 IC50 = 20 nM T61746 C7Y4QZ 44430104 IC50 = 606 nM T61746 C3ICA4 44430105 IC50 = 770 nM T61746 CYX6D9 44430106 IC50 = 205 nM T61746 CX2YD8 44430109 IC50 = 436 nM T61746 C7MCA8 44438028 Ki = 2200 nM T61746 CVD7L4 44442257 IC50 > 10000 nM T61746 CX15UA 44444919 IC50 > 30000 nM T61746 CUXF67 44444920 IC50 > 30000 nM T61746 C1DHA5 44444921 IC50 > 30000 nM T61746 CJWB56 44444922 IC50 > 30000 nM T61746 C0NB8D 44444923 IC50 > 30000 nM T61746 C9P7OQ 44444924 IC50 > 30000 nM T61746 CXO56L 44447657 IC50 > 10000 nM T61746 CB6H5U 44447658 IC50 > 10000 nM T61746 C1U6JA 44447659 IC50 > 10000 nM T61746 CV3T1A 44447660 IC50 > 10000 nM T61746 CF7AV1 44447661 IC50 > 10000 nM T61746 C7HRP2 44447662 IC50 > 10000 nM T61746 C0CZ7P 44447663 IC50 = 100 nM T61746 CAF54M 44447664 IC50 = 1528 nM T61746 CC4J7S 44447665 IC50 = 434 nM T61746 C7QW0F 44449893 IC50 = 22000 nM T61746 CW30VS 44449926 IC50 = 6000 nM T61746 C40EDY 44449928 IC50 = 4500 nM T61746 C83KAR 44449929 IC50 = 4900 nM T61746 C59IFW 44449957 IC50 = 3000 nM T61746 CH7YE8 44449958 IC50 = 1800 nM T61746 CTQ3A1 44449959 IC50 = 1700 nM T61746 CF59ZH 44449960 IC50 = 3300 nM T61746 C59OXW 44449989 IC50 = 210 nM T61746 C69NRS 44449990 IC50 = 300 nM T61746 CC0AG3 44452909 Ki = 90 nM T61746 CB8IX2 44452912 Ki = 7000 nM T61746 CXJF30 44452936 Ki = 2100 nM T61746 CVCJ36 44452938 Ki = 2 nM T61746 C4ZBF6 44452963 Ki = 34000 nM T61746 CWCK10 44452964 Ki = 16000 nM T61746 CF9PC3 44452965 Ki = 25000 nM T61746 C5I2XF 44457308 Ki = 5900 nM T61746 C86ORE 44459987 IC50 = 10000 nM T61746 CG8N9C 44462242 Ki = 4560 nM T61746 C37WKU 44464160 IC50 > 100000 nM T61746 C9TFJ8 44464926 IC50 = 12589.25 nM T61746 CYO0T1 44465454 IC50 = 6309.57 nM T61746 CE83YL 44465721 IC50 = 1584.89 nM T61746 CVD48M 44478848 IC50 = 40 nM T61746 CJR45G 44479122 IC50 = 32 nM T61746 C8I9QK 44479381 IC50 = 110 nM T61746 CWS3K7 44479385 IC50 = 32 nM T61746 C2PK4G 44479635 IC50 = 23 nM T61746 CB73NC 44479637 IC50 = 11 nM T61746 CA48JP 44480468 IC50 > 15000 nM T61746 C0ZE3C 44480469 IC50 > 15000 nM T61746 C0G5ET 44480470 IC50 > 50000 nM T61746 CH7I8C 44480471 IC50 > 15000 nM T61746 CPDQ74 44480723 IC50 > 15000 nM T61746 CPN9C7 44480724 IC50 > 50000 nM T61746 CZ62AB 44480725 IC50 > 50000 nM T61746 C8SL0N 44480726 IC50 > 15000 nM T61746 C1ZOM7 44480727 IC50 = 2500 nM T61746 CZE95Q 44480728 IC50 = 4000 nM T61746 CYBH29 44480974 IC50 > 15000 nM T61746 CA0F2M 44480975 IC50 = 13000 nM T61746 CFJ21O 44480976 IC50 > 15000 nM T61746 C94NWI 44480977 IC50 > 15000 nM T61746 CFE2H6 44480978 IC50 = 8400 nM T61746 COJ38W 44480979 IC50 > 50000 nM T61746 C45EMI 44481231 IC50 > 15000 nM T61746 COL4C2 44481232 IC50 > 15000 nM T61746 CJ1M6E 44481233 IC50 > 50000 nM T61746 C32YDM 44481234 IC50 > 50000 nM T61746 CG1X4W 44481235 IC50 > 50000 nM T61746 CG5YU6 44481236 IC50 > 50000 nM T61746 CUHM64 44481503 IC50 > 50000 nM T61746 CBGO51 44481504 IC50 = 4700 nM T61746 CT9W2X 44481505 IC50 = 8600 nM T61746 C1S0KC 44481506 IC50 = 3900 nM T61746 CRQ32O 44481507 IC50 = 13000 nM T61746 C1E6AT 44481508 IC50 > 50000 nM T61746 CCW6N4 44481776 IC50 > 50000 nM T61746 CCOK78 44481777 IC50 > 15000 nM T61746 CK1E7H 44481778 IC50 > 15000 nM T61746 CFYP92 44482496 IC50 = 38 nM T61746 C1LWX5 44552274 Ki = 3300 nM T61746 CIP6M8 44552275 Ki = 7500 nM T61746 CWJV95 44552368 Ki = 16700 nM T61746 C9UGD8 44562096 Ki = 2910 nM T61746 CV1IL5 44565796 IC50 > 10000 nM T61746 CLH74F 44565900 IC50 = 1640 nM T61746 CMIP10 44565901 IC50 = 1530 nM T61746 C70BXJ 44565925 IC50 = 1750 nM T61746 CS6YO0 44566187 IC50 = 14.2 nM T61746 CSF17Z 44566188 IC50 = 3.11 nM T61746 CJP3U5 44566195 IC50 = 396.8 nM T61746 CUFJ57 44566196 IC50 = 12690 nM T61746 C8YPA6 44572419 Ki = 6400 nM T61746 C3L7IV 44572420 Ki = 13700 nM T61746 CFZ3L7 44572422 Ki = 850 nM T61746 CFZB79 44572423 Ki = 7300 nM T61746 CGC0W5 44572424 Ki = 9900 nM T61746 CP1HU3 44580453 Ki = 244000 nM T61746 CU80NJ 44580454 Ki = 94000 nM T61746 C7D3CY 44580455 Ki = 1018000 nM T61746 CX40GW 46226591 Ki = 4000 nM T61746 C8HEC4 46226622 Ki = 6700 nM T61746 CELQ42 46226646 Ki = 16300 nM T61746 CA7V4F 46226655 Ki = 3700 nM T61746 C4YAJ7 46228924 IC50 > 10000000 nM T61746 CD1W6B 46232382 IC50 > 10000 nM T61746 CRYZ16 46232383 IC50 > 10000 nM T61746 C60TNV 46232384 IC50 > 10000 nM T61746 C1I8LN 46232385 IC50 > 10000 nM T61746 C4P7CD 46232387 IC50 > 10000 nM T61746 CQN2I7 46232805 IC50 > 10000 nM T61746 C39QNG 46232806 IC50 > 10000 nM T61746 CFW92U 46232807 IC50 > 10000 nM T61746 CWD0B5 46232808 IC50 > 10000 nM T61746 CPB62W 46232809 IC50 > 10000 nM T61746 CU8ZB6 46232845 IC50 > 10000 nM T61746 C32ENI 46232846 IC50 > 10000 nM T61746 CX0O3T 46232848 IC50 > 10000 nM T61746 C0WJ4R 46232849 IC50 > 10000 nM T61746 CU5KA6 46232850 IC50 > 10000 nM T61746 C5W2SX 46232966 IC50 > 10000 nM T61746 CEJ0Z8 46232968 IC50 > 10000 nM T61746 C60SCN 46232969 IC50 > 10000 nM T61746 CL6GY7 46232970 IC50 > 10000 nM T61746 CA9QH7 46232971 IC50 > 10000 nM T61746 C8N2YC 46233007 IC50 = 1590 nM T61746 C8HR1S 46233008 IC50 > 10000 nM T61746 CY84AW 46233009 IC50 > 10000 nM T61746 CRS52G 46233010 IC50 > 10000 nM T61746 CC64UL 46233011 IC50 > 10000 nM T61746 C0U9OQ 46233012 IC50 > 10000 nM T61746 CV74LQ 46233041 IC50 > 10000 nM T61746 C1ZG2T 46233042 IC50 > 10000 nM T61746 C6IJO8 46233043 IC50 > 10000 nM T61746 CZ1E0U 46233044 IC50 > 10000 nM T61746 CH29YW 46233045 IC50 > 10000 nM T61746 CO94IL 46233046 IC50 > 10000 nM T61746 COEI67 46233047 IC50 > 10000 nM T61746 CR80PA 46237233 Ki > 330 nM T61746 CC2N0F 46842579 IC50 > 10000 nM T61746 CV6SW4 46842581 IC50 > 10000 nM T61746 CM2D1G 46842582 IC50 > 10000 nM T61746 CIU1R5 46842626 IC50 > 10000 nM T61746 C37OSC 46842709 IC50 > 10000 nM T61746 C6HD4M 46865101 IC50 > 10000 nM T61746 CC7DG3 46866398 IC50 = 6457 nM T61746 CGT1Z2 46881448 IC50 > 10000 nM T61746 CH9ON3 46881449 IC50 > 10000 nM T61746 CF15KQ 46881450 IC50 > 10000 nM T61746 CN58BG 46882092 IC50 > 10000 nM T61746 CG9X3C 46882094 IC50 > 10000 nM T61746 CZ5KP8 46882095 IC50 > 10000 nM T61746 CPQZ83 46882096 IC50 > 10000 nM T61746 CUI91D 46905615 IC50 > 3000 nM T61746 C3XS0I 46930720 Ki = 750 nM T61746 CTE76C 46930722 Ki = 2340 nM T61746 C3F4XK 46930810 Ki = 440 nM T61746 CJ59AN 46930811 Ki = 111000 nM T61746 CLV0F9 46930812 Ki = 75500 nM T61746 CZR16J 46930813 Ki = 475000 nM T61746 CFWU08 46946224 IC50 > 25000 nM T61746 CVT40A 46947220 IC50 = 47600 nM T61746 CAFW31 49783666 IC50 > 10000 nM T61746 CI7P2B 49797571 IC50 > 50000 nM T61746 CI59MV 49797572 IC50 > 50000 nM T61746 C96CKU 49797573 IC50 > 50000 nM T61746 C9LNK5 49798881 Ki > 150000 nM T61746 CE6Z7V 49798882 Ki = 10900 nM T61746 C5CY7U 49798883 Ki = 2230 nM T61746 C3B8FE 49798886 Ki = 25000 nM T61746 C8R6CQ 49798901 Ki = 20400 nM T61746 C7YZV2 49798902 Ki = 12400 nM T61746 CO7I0B 49798903 Ki = 13700 nM T61746 CVT4U3 49798904 Ki = 39100 nM T61746 C3Y6OC 49798905 Ki = 6100 nM T61746 C4NB3R 49834903 IC50 = 3600 nM T61746 CQ3W9J 49834904 IC50 = 5700 nM T61746 CX1WU8 49834905 IC50 = 13300 nM T61746 CA96LF 49834906 IC50 = 63300 nM T61746 CB9MS2 49834907 IC50 = 3200 nM T61746 C74RAF 49834908 IC50 = 13100 nM T61746 CN8E2A 49834971 IC50 = 700 nM T61746 COG9T6 49834972 IC50 = 38000 nM T61746 CGPM91 49834975 IC50 = 7100 nM T61746 CJ73DH 49835032 IC50 = 39400 nM T61746 C8XR4Q 49835033 IC50 = 6400 nM T61746 CXE51M 49835035 IC50 = 22900 nM T61746 CKRG17 49835144 IC50 > 25000 nM T61746 C9NO4U 49835145 IC50 > 25000 nM T61746 CP4S5A 49835673 IC50 = 6200 nM T61746 CS3HC6 49835674 IC50 = 8500 nM T61746 C8O3UF 49835732 IC50 = 29700 nM T61746 C37RZT 49862146 IC50 > 10000 nM T61746 CJ0HY8 49862186 IC50 > 10000 nM T61746 CKA53W 49862308 IC50 > 10000 nM T61746 C8B2WE 49862309 IC50 > 10000 nM T61746 CR13LF 49862310 IC50 > 10000 nM T61746 C38BJK 49862365 IC50 > 10000 nM T61746 C1Z9VQ 49862366 IC50 > 10000 nM T61746 C6W1UJ 49862367 IC50 > 10000 nM T61746 CIFP19 49862368 IC50 > 10000 nM T61746 CMW23V 49862369 IC50 > 10000 nM T61746 CI4J0A 49862370 IC50 > 10000 nM T61746 C1XBM6 49862420 IC50 > 10000 nM T61746 CKV06S 49862421 IC50 > 10000 nM T61746 CN4GD6 49862422 IC50 > 10000 nM T61746 CA7K8Q 49862423 IC50 > 10000 nM T61746 CS92IZ 49862471 IC50 > 10000 nM T61746 C1NAQ5 49862472 IC50 > 10000 nM T61746 C5OD6J 49862473 IC50 > 10000 nM T61746 CFCH31 49862474 IC50 > 10000 nM T61746 C29OGE 49862475 IC50 > 10000 nM T61746 CVOG15 49865938 Ki > 100000 nM T61746 CRI85M 50898446 IC50 = 1600 nM T61746 C18RNG 50925386 Ki = 510 nM T61746 C4I0JY 50925524 IC50 = 383 nM T61746 C01DJG 50993971 Ki = 840 nM T61746 CW9X3R 50993972 Ki = 55 nM T61746 CIC7H1 50993973 Ki = 4.3 nM T61746 C3UB9Y 50993974 Ki = 0.88 nM T61746 CMS13V 50994055 Ki = 0.48 nM T61746 CPT6I5 50994056 Ki = 0.38 nM T61746 CB4X6Y 50994057 Ki = 1.3 nM T61746 CSY4W0 50994058 Ki = 0.65 nM T61746 CQ08HC 50994059 Ki = 2.8 nM T61746 C30WKN 50994060 Ki = 1.3 nM T61746 C8A1GN 50994137 Ki = 2.4 nM T61746 C6K3EJ 50994138 Ki = 2.4 nM T61746 CN6ZM0 50994139 Ki > 330 nM T61746 CF7SN9 50994140 Ki > 330 nM T61746 CU7M1P 50994141 Ki > 22000 nM T61746 C4FE0T 50994142 Ki = 0.36 nM T61746 C96FHG 51033722 IC50 = 1424 nM T61746 C8FM4W 52940769 Ki = 1420 nM T61746 C4JB5S 52941092 IC50 > 10000 nM T61746 CDC64G 52941172 IC50 > 10000 nM T61746 C7DO0F 52941283 IC50 = 68 nM T61746 CU1TW6 52941414 IC50 = 577 nM T61746 C71VFU 52941469 IC50 = 5754 nM T61746 C8BP5L 52941833 IC50 > 10000 nM T61746 CQ39TK 52941839 IC50 > 10000 nM T61746 CDO45C 52941841 IC50 > 10000 nM T61746 CW05MV 52942797 IC50 = 3236 nM T61746 C9MK7J 52942931 IC50 = 312 nM T61746 CVO3U2 52943063 IC50 > 10000 nM T61746 C2AV9H 52943244 IC50 > 10000 nM T61746 CYLF86 52943307 IC50 > 10000 nM T61746 CQDG96 52943578 IC50 > 10000 nM T61746 C4TY6S 52943722 IC50 > 10000 nM T61746 CQ6N0I 52943841 IC50 > 10000 nM T61746 C9B6DJ 52944285 IC50 > 10000 nM T61746 C1UP6N 52945298 IC50 > 10000 nM T61746 CF1LS6 52945475 IC50 > 10000 nM T61746 CN6V0H 52945759 IC50 > 10000 nM T61746 CV8L9Z 52945985 IC50 = 59 nM T61746 CLJ83U 52946267 IC50 = 397 nM T61746 CBD6S0 52946687 IC50 > 10000 nM T61746 CS2NX6 52946690 IC50 > 10000 nM T61746 CND9C6 52947170 IC50 > 10000 nM T61746 CT28XU 52947761 IC50 = 668 nM T61746 CI0S1W 52947952 IC50 > 10000 nM T61746 C75SHQ 52948860 IC50 = 15136 nM T61746 C7SJ1Y 53304087 IC50 = 378 nM T61746 C56OCA 53317528 IC50 = 5011.87 nM T61746 CM60RJ 53317530 IC50 > 25118.86 nM T61746 C5A6IH 53317737 IC50 = 1258.93 nM T61746 C6FEH9 53318816 IC50 > 25118.86 nM T61746 CJAX07 53318817 IC50 > 25118.86 nM T61746 CG5AP6 53318818 IC50 > 25118.86 nM T61746 CJ3PN0 53319501 IC50 > 10000 nM T61746 C7V2DA 53322116 IC50 > 10000 nM T61746 CQ8O1R 53322117 IC50 > 10000 nM T61746 C0QV5D 53322753 IC50 = 3981.07 nM T61746 CHB96K 53324300 IC50 = 10000 nM T61746 CR1L4Y 53325394 IC50 > 25118.86 nM T61746 CVU0J1 53326656 IC50 = 3981.07 nM T61746 C4OP3N 53328398 IC50 > 2500 nM T61746 CKH9C7 53328587 IC50 = 417 nM T61746 CIMR05 54578483 Ki = 3600 nM T61746 CX58ZH 54578708 Ki = 4500 nM T61746 C84WMD 54578709 Ki = 2500 nM T61746 CK74GM 54579405 Ki = 3300 nM T61746 CY0WE3 54768945 Ki = 13000 nM T61746 C0RFL5 54768946 Ki = 10300 nM T61746 C82FCG 54768947 Ki = 9000 nM T61746 CM4YE2 54768948 Ki = 7400 nM T61746 CJ67EC 54768949 Ki = 13800 nM T61746 CXA98K 54768950 Ki = 6000 nM T61746 C7XZ9Y 54769181 Ki = 3300 nM T61746 C3YVZ9 54769182 Ki = 4000 nM T61746 C96HPC 54769183 Ki = 10500 nM T61746 C75WBG 54769184 Ki = 9100 nM T61746 C48EJD 54769407 Ki = 10800 nM T61746 C3J1KQ 54769408 Ki = 9700 nM T61746 CE3TV0 54769409 Ki = 97100 nM T61746 CQ08JC 54769410 Ki = 49400 nM T61746 CDL43S 54769411 Ki = 14800 nM T61746 C3AC1Y 54769412 Ki = 51600 nM T61746 CDI34B 54769413 Ki = 351000 nM T61746 C19TGW 54769414 Ki = 28300 nM T61746 C2VT4I 54769628 Ki = 10130 nM T61746 C2GZ8P 54769629 Ki = 8950 nM T61746 C1NJ6T 56654510 Ki > 330 nM T61746 CDAN29 56657787 IC50 = 460 nM T61746 CU26MD 56657788 IC50 = 23 nM T61746 CD5W7V 56661312 IC50 = 370 nM T61746 CIX1H6 56664780 IC50 = 270 nM T61746 C24ZAM 56664781 IC50 = 220 nM T61746 C24PVH 56664782 IC50 = 270 nM T61746 C70CMI 56664783 IC50 = 530 nM T61746 CB57PR 56668196 IC50 = 410 nM T61746 CU59KM 56671669 IC50 = 310 nM T61746 C46EFG 56675090 IC50 = 52 nM T61746 CDN7E0 56675091 IC50 = 440 nM T61746 CX0FH5 56678398 IC50 = 580 nM T61746 C3WEQ5 56678399 IC50 = 1500 nM T61746 CD67LW 56678400 IC50 = 110 nM T61746 CLQ5N8 56680462 Ki = 4400 nM T61746 CT2M3V 56947698 IC50 = 1800 nM T61746 CT0PC4 56947827 IC50 = 6600 nM T61746 CA9LP1 56948072 IC50 = 2400 nM T61746 CTS0D3 57394400 Ki = 500 nM T61746 C84CHB 57541268 IC50 > 2900 nM T61746 CK5X0U 57619789 IC50 > 10000 nM T61746 CH3M0B 59543520 IC50 > 25000 nM T61746 CCR9Q8 59543629 IC50 = 14900 nM T61746 C3ESJ1 59543757 IC50 = 35200 nM T61746 CZV45P 59619390 IC50 > 25000 nM T61746 CLX2Y4 60148518 Ki = 24000 nM T61746 C0DA6M 60166364 Ki = 40000 nM T61746 C4G1SF 60166365 Ki = 24000 nM T61746 COM7U3 60166366 Ki = 5100 nM T61746 COQ82A 60166367 Ki = 6400 nM T61746 C2Y7EK 60166492 Ki = 5400 nM T61746 C4PHR1 60166493 Ki = 34000 nM T61746 CG4DZ7 60166494 Ki = 3900 nM T61746 C5E2PB 60166495 Ki = 3400 nM T61746 CXD39V 60166496 Ki = 6800 nM T61746 CM8XO5 60166497 Ki = 7200 nM T61746 CA95CZ 60195809 IC50 = 9820 nM T61746 CY3VC4 60195810 IC50 = 8750 nM T61746 CVRJ91 60195812 IC50 = 712 nM T61746 CE6AH0 60195813 IC50 = 7630 nM T61746 C8ILH6 60195902 IC50 = 455 nM T61746 CX4N2V 60195903 IC50 = 1420 nM T61746 C4PQ6E 60195904 IC50 = 44900 nM T61746 CNUI89 60195905 IC50 = 73500 nM T61746 C23JUZ 60195906 IC50 = 31200 nM T61746 CM9V8X 67950125 IC50 = 58000 nM T61746 C7D1ZU 67950129 IC50 > 200000 nM T61746 CC4V3N 67950186 IC50 = 33000 nM T61746 CDN75Y 67950205 IC50 = 29000 nM T61746 CJ5YT6 67971215 IC50 = 10000 nM T61746 CGMR05 67971930 IC50 = 110000 nM T61746 CB85MH 68304447 IC50 = 16 nM T61746 C3E9JI 68304452 IC50 = 544 nM T61746 CB1SY9 68304484 IC50 = 231 nM T61746 CBY9R7 68304488 IC50 > 2500 nM T61746 C3RIC7 68304489 IC50 = 511 nM T61746 CK51WZ 68304496 IC50 = 20 nM T61746 C4U6HZ 68304619 IC50 > 2500 nM T61746 C8UVT5 68304620 IC50 = 721 nM T61746 C8AO7C 68305368 IC50 = 984 nM T61746 CF2P9S 68305374 IC50 = 459 nM T61746 C8L1ER 68305392 IC50 = 429 nM T61746 CVYU02 68305409 IC50 = 81 nM T61746 C7L6PO 68305417 IC50 = 67 nM T61746 C3AN0E 68305418 IC50 = 242 nM T61746 CDT73A 68305425 IC50 = 88 nM T61746 C2V1GR 68305444 IC50 = 3571 nM T61746 C79MJP 68305510 IC50 > 2500 nM T61746 CC0Z8M 68305511 IC50 = 540 nM T61746 C1MZ3P 68305513 IC50 = 494 nM T61746 CQ2T5X 68305514 IC50 = 446 nM T61746 CEHD91 68305517 IC50 = 3404 nM T61746 C4MC0T 68305519 IC50 = 512 nM T61746 CS9NW1 68305525 IC50 = 628 nM T61746 CH2TE0 68305538 IC50 = 283 nM T61746 C4CDR6 68305546 IC50 = 50 nM T61746 C0OV9J 68305563 IC50 = 2847 nM T61746 CDUY03 68305567 IC50 = 3049 nM T61746 CU17ZJ 68305595 IC50 > 2500 nM T61746 CKPD91 69224014 Ki = 85000 nM T61746 CSF35K 70274227 IC50 = 977 nM T61746 CI0XF8 70274815 IC50 = 5011.87 nM T61746 CXT5G7 70275845 IC50 = 3430 nM T61746 C5P3BO 70275923 IC50 = 24900 nM T61746 C3U9IH 70276243 IC50 = 3981.07 nM T61746 CCG16F 70276365 IC50 = 5011.87 nM T61746 C0T3LC 70276605 IC50 = 3060 nM T61746 CE1J0O 70276811 IC50 = 5011.87 nM T61746 C06WFN 70276830 IC50 = 25118.86 nM T61746 CDQ85E 70276990 IC50 = 7943.28 nM T61746 CGET13 70278898 IC50 = 1000 nM T61746 C2GT5H 70280758 IC50 = 3162.28 nM T61746 CI53XU 70281040 IC50 = 3510 nM T61746 CA6DM2 70281073 IC50 = 2511.89 nM T61746 CJQX06 70681840 IC50 = 102000 nM T61746 CW8L0K 70682252 IC50 > 10000 nM T61746 C1UIK4 70682253 IC50 > 10000 nM T61746 CSW1R7 70682254 IC50 > 10000 nM T61746 CY2WE3 70682255 IC50 > 10000 nM T61746 CVHX94 70682256 IC50 > 10000 nM T61746 CNF23Q 70682257 IC50 > 10000 nM T61746 CZ84UX 70682584 IC50 = 3981.07 nM T61746 CR45PO 70683941 IC50 = 5300 nM T61746 C8S1DB 70684341 IC50 > 10000 nM T61746 CH7L2N 70684342 IC50 > 10000 nM T61746 CM2V0E 70686501 IC50 > 10000 nM T61746 CSPH68 70686502 IC50 > 10000 nM T61746 CL9RE3 70686820 IC50 = 3162.28 nM T61746 C65EDY 70686822 IC50 = 2511.89 nM T61746 CWE9C8 70688597 IC50 > 10000 nM T61746 CV20NB 70688598 IC50 > 10000 nM T61746 CJ4FO1 70688599 IC50 > 10000 nM T61746 CIR23C 70688600 IC50 > 10000 nM T61746 C5NMF8 70688601 IC50 > 10000 nM T61746 C5IYR0 70688897 IC50 = 2511.89 nM T61746 CA1Q0F 70690660 IC50 > 10000 nM T61746 CZY5R0 70690661 IC50 > 10000 nM T61746 C2Z8JP 70690662 IC50 > 10000 nM T61746 C73CZT 70690663 IC50 > 10000 nM T61746 C2H1NL 70690664 IC50 > 10000 nM T61746 CE8Q4U 70692809 IC50 > 10000 nM T61746 CND37B 70692810 IC50 > 10000 nM T61746 CZOF81 70693115 IC50 = 3162.28 nM T61746 CMFW03 70693116 IC50 = 6309.57 nM T61746 C5RSJ0 70693117 IC50 = 3981.07 nM T61746 C36JBX 70694841 IC50 > 10000 nM T61746 C86ETZ 70694842 IC50 > 10000 nM T61746 CAU9C4 70694843 IC50 > 10000 nM T61746 C4A7HL 70694844 IC50 > 10000 nM T61746 C01IDC 70695171 IC50 = 3162.28 nM T61746 CURI37 70696209 Ki = 1.58 nM T61746 C8HEM6 70696892 IC50 > 10000 nM T61746 CK5RP0 70696893 IC50 > 10000 nM T61746 C34WHG 70697225 IC50 = 5011.87 nM T61746 C1SD3A 70701946 Ki > 330 nM T61746 C0H1BV 70788951 IC50 = 250000 nM T61746 C0MNY4 71127989 IC50 = 532 nM T61746 C3T2UW 71135835 IC50 = 367 nM T61746 CUB38S 71449749 IC50 > 2900 nM T61746 C08LGJ 71451733 IC50 = 315 nM T61746 CI7Z8B 71451734 IC50 = 645 nM T61746 C7RJG8 71453558 IC50 = 572 nM T61746 CDR10X 71453560 IC50 = 1440 nM T61746 CPGT63 71454020 Ki > 40000 nM T61746 CFUS41 71455276 IC50 = 1180 nM T61746 CUQL74 71455277 IC50 = 2940 nM T61746 C0KUW5 71455278 IC50 = 1690 nM T61746 C7Z0HF 71455279 IC50 = 649 nM T61746 CU48QH 71455759 Ki > 40000 nM T61746 C9YJG7 71457065 IC50 = 1270 nM T61746 CK7ZF4 71458275 EC50 = 700 nM T61746 C1UOK5 71458276 EC50 = 200 nM T61746 CCH47M 71458921 IC50 = 1440 nM T61746 CP7MZ5 71458922 IC50 = 971 nM T61746 CCA46N 71458923 IC50 = 1850 nM T61746 CQT1C2 71458924 IC50 = 462 nM T61746 C6RZF3 71459429 Ki = 140 nM T61746 CDW0I7 71460731 IC50 = 399 nM T61746 CL6Y4C 71460733 IC50 = 603 nM T61746 CC2OF7 71520320 Ki = 58000 nM T61746 C7JNE5 71520321 Ki = 82000 nM T61746 CKI54R 71520322 Ki = 8000 nM T61746 CF52NJ 71520323 Ki = 76000 nM T61746 CZM3L7 71520324 Ki = 5000 nM T61746 CL10QN 71520325 Ki = 116000 nM T61746 CF0V4Y 71520326 Ki = 87000 nM T61746 CA2D9X 71520327 Ki = 74000 nM T61746 CGA61K 71520445 Ki = 125000 nM T61746 CRE8Q0 71520446 Ki = 117000 nM T61746 C74IMH 71521815 Ki = 171000 nM T61746 CLU89M 71521816 Ki = 94000 nM T61746 C5YQ6V 71602930 IC50 > 10000 nM T61746 CY7EL9 71602931 IC50 > 10000 nM T61746 CC61PX 71602932 IC50 > 10000 nM T61746 CH5QG3 71602933 IC50 > 10000 nM T61746 COU6R5 71602979 IC50 > 10000 nM T61746 CR6JV1 71602981 IC50 > 10000 nM T61746 CP87FL 71602983 IC50 > 10000 nM T61746 C34RLW 71602984 IC50 > 10000 nM T61746 CL6B0E 71602986 IC50 > 10000 nM T61746 CQ1ZN0 71603042 IC50 > 10000 nM T61746 C6SWY5 71603043 IC50 > 10000 nM T61746 CD0Z4V 71603045 IC50 > 10000 nM T61746 C1YCF7 71603046 IC50 > 10000 nM T61746 C2VH5F 71603047 IC50 > 10000 nM T61746 CQ76CG 71603106 IC50 > 10000 nM T61746 CF9J1B 71603109 IC50 > 10000 nM T61746 CMSE93 71603111 IC50 > 10000 nM T61746 CIU41Z 71603112 IC50 > 10000 nM T61746 C9GMP4 71603168 IC50 > 10000 nM T61746 CSI94H 71612693 Ki = 113000 nM T61746 CH65CP 71612694 Ki = 74000 nM T61746 CER82H 71612695 Ki = 39000 nM T61746 C3WV1B 71612696 Ki = 312000 nM T61746 CJ71KZ 71612697 Ki = 3387000 nM T61746 COZ0E4 71612901 Ki = 84000 nM T61746 CQ3XD4 71612902 Ki = 301000 nM T61746 C4U0TK 71612903 Ki = 26000 nM T61746 CA82UN 71612904 Ki = 261000 nM T61746 CY02ME 71612905 Ki = 1020000 nM T61746 C4TG6P 71612906 Ki = 706000 nM T61746 C3PY2W 71613098 Ki = 1757000 nM T61746 C7KF1W 71613099 Ki = 134000 nM T61746 CAG6F9 71613100 Ki = 80000 nM T61746 CI0Q7G 71613101 Ki = 148000 nM T61746 CTH19S 71613102 Ki = 860000 nM T61746 CV60XA 71613103 Ki = 51000 nM T61746 C90OHP 71613322 Ki = 623000 nM T61746 CRP54C 71613323 Ki = 2035000 nM T61746 C85WJH 71613324 Ki = 135000 nM T61746 C6HK4W 71615678 Ki = 77000 nM T61746 C7CN4G 71615679 Ki = 38000 nM T61746 C8JN2W 71615680 Ki = 58000 nM T61746 CN32FZ 71615681 Ki = 389000 nM T61746 C4XUV9 71615682 Ki = 245000 nM T61746 C5NV8E 71624115 IC50 > 10000 nM T61746 C8DZ6U 71624118 IC50 > 10000 nM T61746 C8SGK6 71624246 IC50 > 10000 nM T61746 CM64QD 71624362 IC50 > 10000 nM T61746 CK64NT 71624363 IC50 > 10000 nM T61746 CNZ0K4 71624621 IC50 > 100000 nM T61746 C9QY7K 71624622 IC50 > 100000 nM T61746 C0S6HT 71624732 IC50 > 100000 nM T61746 C3CRY6 71624733 IC50 = 95090 nM T61746 C37EVT 71624734 IC50 = 46810 nM T61746 C9P1QH 71624735 IC50 > 100000 nM T61746 CNCX24 71624736 IC50 = 28670 nM T61746 CAN6X5 71656574 IC50 = 9000 nM T61746 CQL6S2 71659902 Ki = 86000 nM T61746 CI6VO9 71716098 Ki = 175000 nM T61746 C63ROI 71717313 Ki = 24000 nM T61746 CB4VU9 71720364 Ki = 36000 nM T61746 C0O5NF 71726670 IC50 > 10000 nM T61746 CW16QR 71738813 IC50 > 10000 nM T61746 CS31TK 71738883 IC50 > 10000 nM T61746 C8ITL0 73107490 Ki = 8000 nM T61746 C7BKZ5 73345448 IC50 = 172000 nM T61746 CIO7K3 73345851 Ki = 2787000 nM T61746 CY1IU2 73345852 Ki = 835000 nM T61746 CDQP51 73347119 Ki = 10000 nM T61746 CJQE58 73348851 Ki = 3406000 nM T61746 C5XOV2 73348852 Ki = 1734000 nM T61746 C31JUR 73348857 Ki = 1303000 nM T61746 C95BEA 73348858 Ki = 1494000 nM T61746 COF4E6 73349875 IC50 > 10000 nM T61746 CM3PH8 73350210 Ki = 7300 nM T61746 CZN1M9 73350437 Ki = 2460000 nM T61746 CMD57T 73350441 Ki = 3545000 nM T61746 CO01PD 73351555 IC50 = 100000 nM T61746 CAYM96 73351955 Ki = 1185000 nM T61746 CMN72X 73352839 IC50 = 8700 nM T61746 C7BYL1 73353012 IC50 > 1000000 nM T61746 C84NFB 73353013 IC50 = 416000 nM T61746 CXR1B9 73353408 Ki = 135000 nM T61746 CNQA65 73354924 Ki = 1547000 nM T61746 C37HIQ 73354926 Ki = 56000 nM T61746 CY81IS 73356107 IC50 > 1000000 nM T61746 CJ6CQ1 73356205 Ki = 7300 nM T61746 CL37SD 73356439 IC50 > 10000 nM T61746 CYSR74 73356489 Ki = 100000 nM T61746 CW9NU4 73895627 Ki = 72 nM T61746 C76KAG 73896141 Ki > 330 nM T61746 CGP83V 78108657 Ki = 2 nM T61746 C4JYM8 78108695 Ki = 5 nM T61746 CWSM27 78108714 Ki = 0.69 nM T61746 CQ8BA7 86140660 Ki = 68000 nM T61746 CZH08W 86635877 IC50 = 2000 nM T61746 CR05TU 89809888 IC50 > 10000 nM T61746 CHJB16 89886996 IC50 > 10000 nM T61746 CIXT20 89888879 IC50 > 10000 nM T61746 C2VJ0N 90644780 Ki > 50000 nM T61746 CEZV52 90644781 Ki = 5000 nM T61746 C5E6BQ 90644782 Ki > 50000 nM T61746 C2ZED8 90644783 Ki > 100000 nM T61746 C68OGA 90644784 Ki > 100000 nM T61746 C0CL3K 90644785 Ki > 50000 nM T61746 CQ2RP1 90644786 Ki = 12070 nM T61746 C8EDQ4 90644787 Ki > 100000 nM T61746 CWB19V 90644788 Ki > 100000 nM T61746 C10MVG 90644789 Ki > 50000 nM T61746 C37YFC 90644790 Ki = 4450 nM T61746 CY0G3V 90644792 Ki > 100000 nM T61746 C4ANR2 90644794 Ki > 100000 nM T61746 C67WRL 90644795 Ki > 50000 nM T61746 CLMJ40 90644796 Ki > 100000 nM T61746 CQ1F6R 90644797 Ki > 100000 nM T61746 CFPT98 90655054 IC50 > 30000 nM T61746 C5JZ8R 90655055 IC50 > 30000 nM T61746 C62SML 90655967 IC50 > 10000 nM T61746 CJ7LT3 90655968 IC50 > 10000 nM T61746 CB61WC 90655969 IC50 > 10000 nM T61746 CIS56R 90663177 Ki = 39000 nM T61746 CU71EO 90663180 Ki = 11000 nM T61746 CX37IK 90663181 Ki = 150 nM T61746 CRY6D3 90663182 Ki = 340 nM T61746 CJ2V9B 90663412 Ki = 15000 nM T61746 C89DWE 90663417 Ki = 560 nM T61746 CX9I6Z 90663418 Ki = 4100 nM T61746 CX7WG9 90665730 Ki = 25000 nM T61746 CFKB46 90665732 Ki = 5000 nM T61746 CB14DH 90665735 Ki = 1350 nM T61746 C0XZH3 90665919 IC50 > 50000 nM T61746 C0HIA4 90665921 IC50 > 50000 nM T61746 C5AIN7 91667613 IC50 > 10000 nM T61746 CGFK60 101201806 IC50 > 30000 nM T61746 CK0AF8 101889645 IC50 = 14900 nM T61746 C7I4XF 101889646 IC50 = 8500 nM T61746 C8E4WS 102323332 IC50 = 2940 nM T61746 CL96MC 102532094 IC50 > 100 ug.mL-1 T61746 CVJF59 118716317 Ki = 3.56 nM T61746 CA79YF 118716318 Ki = 0.459 nM T61746 C3Q5BM 118716319 Ki = 0.406 nM T61746 CI6H0V 118716320 Ki = 194 nM T61746 C5ALU2 118719334 IC50 > 100000 nM T61746 CTE34I 118720232 IC50 > 100000 nM T61746 CSD62B 118720233 IC50 > 100000 nM T61746 C9WF7Q 118720234 IC50 = 8100 nM T61746 C76HIO 118720235 IC50 = 81000 nM T61746 CAT1R6 118720236 IC50 > 100000 nM T61746 CGAF42 118720237 IC50 > 100000 nM T61746 CJ28KZ 118720238 IC50 > 100000 nM T61746 CPH2V9 118720239 IC50 > 100000 nM T61746 CJKA03 118722345 IC50 = 13000 nM T61746 C6I4HX 118722347 IC50 > 200000 nM T61746 C2GV6A 118722348 IC50 = 24000 nM T61746 CRXM26 118722349 IC50 = 58000 nM T61746 CVXD58 118722350 IC50 = 34000 nM T61746 CJ4NR8 118722351 IC50 = 28000 nM T61746 CGXN17 118722352 IC50 = 64000 nM T61746 C1KG8A 118723836 IC50 = 52 nM T61746 CHD0O3 118723838 IC50 = 274 nM T61746 CU4CV8 118723839 IC50 = 311 nM T61746 CZ1M4F 118724181 IC50 > 2500 nM T61746 CMBG29 118724585 IC50 > 100000 nM T61746 C0M3VK 118729722 IC50 > 100 ug.mL-1 T61746 CBD8C5 118729723 IC50 > 100 ug.mL-1 T61746 CTX3W2 118729724 IC50 > 100 ug.mL-1 T61746 CP4D5Q 118729725 IC50 > 100 ug.mL-1 T61746 C0EA2W 118729726 IC50 > 100 ug.mL-1 T61746 CA2P3M 118729727 IC50 > 100 ug.mL-1 T61746 CUC21I 118729728 IC50 > 100 ug.mL-1 T61746 CWU09Y 118729729 IC50 > 100 ug.mL-1 T61746 CLV56Y 118729730 IC50 > 100 ug.mL-1 T61746 C8N5EQ 118729731 IC50 > 100 ug.mL-1 T61746 CH3C4J 118729732 IC50 > 100 ug.mL-1 T61746 CH36VG 122182060 Ki = 41000 nM T61746 CV46XN 122194107 IC50 > 10000 nM T61746 CYO0X5 122194108 IC50 > 10000 nM T61746 CW6K0Z 122194109 IC50 > 10000 nM T61746 CO02XD 122194111 IC50 > 10000 nM T61746 CT51QX 122194112 IC50 > 10000 nM T61746 CYLN40 122194113 IC50 > 10000 nM T61746 CGQ18K 122197351 Ki = 4500 nM T61746 CJSU86 125503087 Ki = 139000 nM T61746 CRS8C6 126610725 IC50 > 10000 nM T61746 CN2IE8 126610758 IC50 > 10000 nM T61746 C2E4BP 126610767 IC50 > 10000 nM T61746 C2HJS3 126610779 IC50 > 10000 nM T61746 C2ZL3O 126610781 IC50 > 10000 nM T61746 CJV56I 126610782 IC50 > 10000 nM T61746 C9QKI3 127020966 IC50 = 200 nM T61746 CV04JO 127037715 IC50 > 50000 nM T61746 CJ27CG 127042051 IC50 > 50000 nM T61746 CAT46D 127042341 IC50 > 50000 nM T61746 C6PIS2 127048500 Ki > 330 nM T61746 CEJ09X 127048537 Ki > 330 nM T61746 CL29KY 127048538 Ki > 330 nM T61746 CD3NX2 127049155 Ki > 330 nM T61746 CFJP85 127049511 Ki > 330 nM T61746 CMT2B9 127049869 Ki = 33000 nM T61746 C14RWJ 127049957 Ki = 630 nM T61746 C8J6DL 127050159 Ki > 330 nM T61746 C43APM 127050163 Ki = 101000 nM T61746 C8VKA5 127050164 Ki = 196000 nM T61746 CZ54XC 127050165 Ki = 26 nM T61746 CI2C3V 127050166 Ki = 19.2 nM T61746 CXM6Z0 127051056 Ki = 3047 nM T61746 CJ7O6G 127051057 Ki = 30345 nM T61746 C6B2ZU 127051058 Ki = 2285 nM T61746 C7V8XZ 127051317 Ki = 132 nM T61746 CSK16Q 127051318 Ki = 368 nM T61746 C7YI4M 127051342 Ki = 126 nM T61746 C6NFU9 127051343 Ki = 120 nM T61746 C6SD7P 127051344 Ki = 1230 nM T61746 CY5CV6 127051345 Ki = 24000 nM T61746 CV14CT 127052305 Ki > 330 nM T61746 COQ94G 127052306 Ki > 330 nM T61746 CG62LJ 127052307 Ki > 330 nM T61746 CIQ79J 127052308 Ki = 330 nM T61746 C8SD2H 134132002 Ki = 6300 nM T61746 C2CT4O 134134083 IC50 = 136 nM T61746 C0U6GR 134134734 Ki = 310 nM T61746 CD5NI4 134134799 Ki = 8 nM T61746 CE53MB 134135884 Ki = 3200 nM T61746 CD0UE9 134136855 IC50 = 34 nM T61746 CW3B7G 134137121 Ki = 710 nM T61746 CF8VA4 134138144 IC50 = 45 nM T61746 C4CT5Z 134139989 Ki = 210 nM T61746 CQ8U5W 134141808 IC50 = 57 nM T61746 C4BXO1 134144535 IC50 = 79 nM T61746 C0YG8C 134148335 IC50 = 57 nM T61746 C4HN8V 134148867 Ki = 68 nM T61746 CH98KJ 134154138 Ki = 34 nM T61746 C2UMT4 134157443 Ki = 310 nM T61746 CUVL51 135872798 IC50 > 10000 nM T61746 CA8Y4C 136002680 IC50 > 10000 nM T61746 CTQY96 136117851 IC50 = 65 nM T61746 CH08TX 136218747 IC50 > 10000 nM T61746 C2DF5Q 136218748 IC50 > 10000 nM T61746 CL46RX 136218749 IC50 > 10000 nM T61746 CGR2E9 136218750 IC50 > 10000 nM T61746 CRUC19 137028456 IC50 > 10000 nM T61746 CR9ZT1 137655120 IC50 = 27 nM T61746 CFQ25D 145967499 IC50 > 5000 nM T61746 CS3T4P 145967500 Ki = 190000 nM T61746 CZ2AL9 145967652 Ki = 102000 nM T61746 CIVB10 145967715 IC50 = 2320 nM T61746 CWLM34 145967735 Ki = 168000 nM T61746 CD8B7F 145967825 Ki = 224000 nM T61746 CHMK10 145967938 Ki = 13000 nM T61746 CLI6T0 145967952 IC50 = 4080 nM T61746 CQ4VH9 145968135 Ki = 171000 nM T61746 CC4AG7 145968405 IC50 > 50000 nM T61746 CDS31M 145968622 IC50 = 1721 nM T61746 C8EJ3C 145968645 Ki = 12000 nM T61746 COB78J 145968830 Ki = 39000 nM T61746 CU6M9N 145968844 Ki = 9000 nM T61746 CE42HR 145968853 Ki = 109000 nM T61746 C1RSP4 145968898 Ki = 96000 nM T61746 C7UW6B 145969091 Ki = 116000 nM T61746 CA40YU 145969275 IC50 = 2210 nM T61746 CN8KP1 145969337 Ki = 32000 nM T61746 CB0Y7Z 145969438 IC50 > 5000 nM T61746 C2WCK0 145969450 IC50 = 2241 nM T61746 CFYH13 145969522 Ki = 22000 nM T61746 CD4T9H 145969728 Ki = 121000 nM T61746 CC0Y7A 145969757 Ki = 128000 nM T61746 CL7KO9 145969878 IC50 = 2371 nM T61746 CTW5P3 145969938 Ki = 94000 nM T61746 C3NAS7 145970030 IC50 = 1270 nM T61746 C8X6JG 145970039 Ki = 124000 nM T61746 CTK40M 145970104 Ki = 18000 nM T61746 CU0RG5 145970355 Ki = 29000 nM T61746 CCGT67 145970471 Ki = 66000 nM T61746 C51ZEH 145970706 Ki = 30000 nM T61746 CJAU37 145970798 Ki = 202000 nM T61746 CS08XI 145970918 IC50 > 5000 nM T61746 C9XKW2 145970931 IC50 = 1104 nM T61746 C50RBK 145971136 Ki = 122000 nM T61746 CXW3F1 145982578 IC50 = 1700 nM T61746 CY7XE4 145982644 IC50 = 5000 nM T61746 C56AXR 145982654 IC50 = 160000 nM T61746 CNC48W 145982661 IC50 = 140 nM T61746 CMS4E9 145982820 IC50 = 50 nM T61746 C7S2TX 145983004 IC50 = 1800 nM T61746 CU5Z9F 145983387 IC50 = 1130 nM T61746 C1OEA0 145983615 IC50 = 70 nM T61746 C6JSW3 145983652 IC50 = 70 nM T61746 C7V2ZF 145983823 IC50 = 1900 nM T61746 CV1A6D 145983891 Ki > 500000 nM T61746 C3JIQ4 145984217 IC50 = 74000 nM T61746 CT8QM9 145984597 IC50 = 32000 nM T61746 C3LH7B 145984676 IC50 = 60 nM T61746 CUT36M 145984739 IC50 = 23900 nM T61746 CJM6L4 145984752 IC50 = 4300 nM T61746 C0BC2Z 145984777 IC50 = 60000 nM T61746 CJK42D 145985003 IC50 = 70 nM T61746 CGC54P 145985016 IC50 = 800 nM T61746 C8AM0K 145985030 Ki = 1400 nM T61746 CURI53 145985037 IC50 = 50 nM T61746 C2LB8K 145985094 IC50 = 11000 nM T61746 CNT63X 145985191 IC50 = 1700 nM T61746 CHCP90 145985556 IC50 = 80 nM T61746 CX6JT1 145985564 IC50 = 10000 nM T61746 CJE7L9 145985615 IC50 = 19000 nM T61746 CL2B3Y 145985677 IC50 = 3500 nM T61746 C9C5YA 145985785 IC50 = 52600 nM T61746 CBK3G5 145985888 IC50 = 90 nM T61746 CQ2RS8 145986120 IC50 = 2300 nM T61746 C6OKB9 145987263 IC50 = 715 nM T61746 COZ6P5 145987960 IC50 > 5000 nM T61746 C7ZCW3 145988622 IC50 > 5000 nM T61746 CN6U8D 145988823 Ki = 8000 nM T61746 C9OAK6 145989037 IC50 = 2500 nM T61746 C87GKT 145989707 IC50 = 2751 nM T61746 C4V2IM 145989709 Ki = 11000 nM T61746 CUAY08 148018738 IC50 = 3000 nM T61746 CQK39B 149491764 IC50 = 3000 nM T61746 C1ZX5D 149494192 IC50 = 3000 nM T61746 CKT12D 155510715 Ki = 6500 nM T61746 CWDS96 155516109 Ki = 64 nM T61746 CO2Y0C 155523098 Ki = 19000 nM T61746 CBN12I 155524050 Ki = 3345 nM T61746 CO3ZF7 155541809 Ki = 37000 nM T61746 C3VR1X 155550446 Ki = 210 nM T61746 CXYT09 155551122 Ki = 909 nM T61746 CCF86H 155553085 Ki = 28000 nM T61746 C2P9GA 155554760 IC50 = 1111 nM T61746 C6O9FK 155556968 Ki = 32000 nM T61746 CQI02B 155559732 Ki > 10000 nM T61746 C8QX2R 155562021 IC50 = 11.9 nM T61746 CFTW36 155567371 Ki = 110 nM T61746 CU42CE 155567829 IC50 = 700 nM T61746 CP5QB8 155568040 IC50 = 300 nM T61746 CHD79T 44408017 IC50 = 35000 nM T61746 CO0N3S 44408050 IC50 = 1800 nM T61746 C58OLD 44517711 IC50 = 3981.07 nM T61746 CT3S1I 44517712 IC50 = 6309.57 nM T61746 CFT38D 45267632 IC50 > 10000 nM T61746 COU83P 45267640 IC50 > 10000 nM T61746 C1U4IF 45267645 IC50 > 10000 nM T61746 CDG5S8 45268499 IC50 = 6309.57 nM T61746 CV8PZ3 45268510 IC50 > 10000 nM T61746 C89ADF 45269361 IC50 = 7943.28 nM T61746 C58PZI 45269375 IC50 > 10000 nM T61746 C5O9EF 45270206 IC50 > 10000 nM T61746 C07ADH 45270207 IC50 > 10000 nM T61746 CVGE81 45270212 IC50 > 10000 nM T61746 C78EXG 45271021 IC50 = 7943.28 nM T61746 C5MBC4 45271038 IC50 > 10000 nM T61746 C65QLD 45271887 IC50 > 10000 nM T61746 CIL8O6 45271888 IC50 = 5011.87 nM T61746 CLFD35 45272742 IC50 = 7943.28 nM T61746 C3WF8S 45272748 IC50 = 6309.57 nM T61746 CQO98K 45272752 IC50 = 6309.57 nM T61746 C9A0IH 45272753 IC50 > 10000 nM T61746 CSYU09 45273681 IC50 > 10000 nM T61746 C0HRW4 70690665 IC50 > 10000 nM T61746 CU60DG 70696894 IC50 > 10000 nM T61746 D00FGA 73737 IC50 = 15000 nM T61746 D00VAN 46232847 IC50 > 10000 nM T61746 D01CSE 52942034 IC50 > 10000 nM T61746 D01NCW 11534772 IC50 = 27000 nM T61746 D03JYN 15722900 IC50 = 13000 nM T61746 D03UYO 44353781 Ki = 370 nM T61746 D04BGT 46881451 IC50 > 10000 nM T61746 D04DFX 136002679 IC50 = 9493 nM T61746 D05MDE 11505372 IC50 = 23000 nM T61746 D05VEV 11556056 IC50 = 1600 nM T61746 D05WZF 10129151 IC50 > 5000 nM T61746 D06FFP 443118 Ki = 150 nM T61746 D06NEB 11693148 IC50 = 850 nM T61746 D06VIP 14774521 Ki > 330 nM T61746 D06WQP 60148519 Ki = 5.8 nM T61746 D07FLB 11637576 Ki > 330 nM T61746 D07FLG 3026 IC50 = 420000 nM T61746 D07RSA 11696652 Ki = 3920 nM T61746 D07ZYE 25195974 Ki = 880 nM T61746 D08KCA 72429 Ki = 5 nM T61746 D08TMM 9851116 IC50 = 5.7 nM T61746 D09AHN 11492732 Ki = 94000 nM T61746 D09FGQ 123985 IC50 = 0.0049 ug.mL-1 T61746 D09GZQ 11713852 IC50 > 150000 nM T61746 D09IMK 11621748 IC50 = 51000 nM T61746 D09NBP 52940642 IC50 > 10000 nM T61746 D0A5WN 11621347 IC50 = 13000 nM T61746 D0A7ER 11514386 Ki > 330 nM T61746 D0A8OV 11086036 Ki > 330 nM T61746 D0B2FE 46882093 IC50 > 10000 nM T61746 D0B2JC 46232967 IC50 = 5690 nM T61746 D0B3US 11585523 IC50 = 140000 nM T61746 D0B4JS 44449925 IC50 > 25000 nM T61746 D0B8TJ 2354 IC50 > 30000 nM T61746 D0D0JU 14849212 Ki = 5940 nM T61746 D0D0LD 9913088 IC50 = 5239 nM T61746 D0G2QG 44343301 IC50 = 460 nM T61746 D0G8OD 11702208 Ki = 32000 nM T61746 D0I0MU 11534625 IC50 = 5800 nM T61746 D0J5VK 67145 IC50 = 90200 nM T61746 D0J7OM 24777047 IC50 > 30000 nM T61746 D0JF8D 11551481 Ki > 330 nM T61746 D0JN8Q 11702265 Ki > 330 nM T61746 D0K0KT 11621207 IC50 = 20000 nM T61746 D0L9VP 5287864 Ki = 64 nM T61746 D0LL1F 52945875 IC50 > 10000 nM T61746 D0M3AP 46232386 IC50 > 10000 nM T61746 D0MD6D 24778186 IC50 > 30000 nM T61746 D0Q4UA 10033311 Ki = 0.088 nM T61746 D0QY3R 11513217 IC50 = 18000 nM T61746 D0RL4S 11714476 IC50 = 41000 nM T61746 D0S4EI 10244468 Ki = 7800 nM T61746 D0T0IR 49865939 Ki = 18900 nM T61746 D0T4FT 46930721 Ki = 1750 nM T61746 D0T7QF 10420833 IC50 = 32000 nM T61746 D0U0XG 11709032 Ki > 330 nM T61746 D0V7LZ 74761 Ki = 15600 nM T61746 D0VE0F 10062714 IC50 = 810 nM T61746 D0X9YD 65036 Ki = 8600 nM T61746 D0Y5IQ 44255320 IC50 = 10000 nM T61746 D0Z0PR 9912381 IC50 = 17 nM T08856 D00MDP 466151 IC50 < 0.4 nM T08856 D0Q8CS 60937 IC50 = 32000 nM T08856 D0S0LZ 54671203 IC50 = 31000 nM T08856 D0VM2L 68740 IC50 = 17600 nM T08856 D05VZE 119031 IC50 = 0.47 nM T08856 D0MW3H 9824350 Ki = 4 nM T08856 D00UCC 9827497 IC50 = 5 nM T08856 D01DVX 9847838 IC50 = 299 nM T08856 D03BOZ 3342298 IC50 = 0.097 nM T08856 D05VNG 9908389 IC50 = 3 nM T08856 D0T9HG 132519 Ki = 0.18 nM T08856 D0Y1XT 128564 Ki = 0.7 nM T08856 CNA81R 1836 IC50 = 81 nM T08856 CYEU83 69033 Ki = 74000 nM T08856 C0PY5N 77754 Ki > 100 nM T08856 CP4O2C 121255 Ki = 69000 nM T08856 C7ROG5 177347 IC50 = 303 nM T08856 CP7Q8T 240910 Ki = 21000 nM T08856 CX3DK6 283995 Ki = 12000 nM T08856 COFX01 352863 Ki = 70000 nM T08856 CK9M3P 445018 IC50 = 6.4 nM T08856 CBTK84 446505 IC50 = 1700 nM T08856 C4D7TS 448002 Ki = 9 nM T08856 CC54LQ 450256 IC50 > 100000 nM T08856 C9I8WB 478379 Ki = 0.4 nM T08856 CN6E3U 2366268 IC50 = 9300 nM T08856 CN62WX 2800809 IC50 = 3000 nM T08856 CY3TD6 3348132 Ki = 2.5 nM T08856 CME24U 3649035 IC50 = 25000 nM T08856 CZBY34 5220706 Ki = 71000 nM T08856 CZS0G5 5276565 IC50 > 100000 nM T08856 C3JN0F 5277465 IC50 = 30000 nM T08856 CRJK67 5277481 IC50 > 100000 nM T08856 CYF7S5 5277490 IC50 > 100000 nM T08856 CJ3QI1 5288814 IC50 = 881 nM T08856 C5IDT0 5289314 Ki = 14 nM T08856 CZC3I7 5326979 IC50 = 1200000 nM T08856 CLVN34 5496618 Ki = 121000 nM T08856 C1LQD2 6540261 Ki = 700 nM T08856 CN5L2B 6852147 Ki = 0.6 nM T08856 CPFV65 6916013 Ki = 126 nM T08856 C0FQW9 7063077 Ki = 275 nM T08856 C7Y1BX 9543420 IC50 = 5.3 nM T08856 CIJ25V 9794947 IC50 > 100000 nM T08856 CLK61C 9797144 Ki = 37 nM T08856 CIXD67 9802768 IC50 = 1.8 nM T08856 C0L5BU 9817358 Ki = 239.88 nM T08856 CTO36D 9817594 IC50 = 50000 nM T08856 C8E2LN 9821077 IC50 = 2 nM T08856 C5OE1B 9821883 Ki = 23 nM T08856 C6KJ9W 9822461 IC50 = 0.81 nM T08856 C6IX7G 9822926 IC50 = 1.2 nM T08856 CL0G8K 9825927 IC50 = 19.95 nM T08856 C1A7NJ 9827355 Ki = 0.39 nM T08856 C7SRM4 9837496 IC50 > 100000 nM T08856 C2R3JP 9842741 IC50 = 1 nM T08856 CE9AL3 9847113 IC50 = 0.9 nM T08856 C4IEK0 9850035 IC50 = 1.9 nM T08856 C5DGI9 9851911 IC50 = 2.4 nM T08856 CI8Z0R 9866250 IC50 = 1.4 nM T08856 CJS23I 9868333 Ki > 3100 nM T08856 CZO2I0 9870133 IC50 = 3 nM T08856 CHU9I8 9871883 IC50 = 1.2 nM T08856 CW8IC4 9882151 IC50 = 1000 nM T08856 C0ZT7A 9883002 Ki = 2100 nM T08856 CZBK85 9886177 IC50 = 130 nM T08856 CD1U5P 9889190 IC50 = 9.4 nM T08856 C6TV1K 9889336 IC50 = 2 nM T08856 CH69LT 9892815 IC50 = 1.7 nM T08856 CSIB97 9896504 IC50 > 30000 nM T08856 C03GVA 9932290 Ki = 230 nM T08856 CDXR37 9933197 IC50 = 9.4 nM T08856 C5E7PR 9933720 Ki = 2 nM T08856 C65ION 9935032 IC50 = 1.3 nM T08856 CG38KL 9936728 Ki = 1.1 nM T08856 CMI06Q 9939403 Ki = 30000 nM T08856 C16HTN 9948666 Ki = 43 nM T08856 COVR98 9951986 IC50 = 20 nM T08856 C9X0YR 9954867 Ki = 171 nM T08856 C32HAZ 9954953 Ki < 2 nM T08856 CK9HX0 9955125 IC50 = 10 nM T08856 C3Q2UJ 9956686 IC50 = 0.4 nM T08856 CN76XI 9957653 IC50 = 1 nM T08856 CHS9L0 9974516 Ki = 240 nM T08856 C0HL2X 9976697 IC50 = 1.4 nM T08856 CA0XP7 9977927 Ki = 400 nM T08856 CJGR30 9983604 IC50 = 1.2 nM T08856 C8W5UK 9999879 IC50 = 228 nM T08856 C6TO0A 10001582 Ki = 1.1 nM T08856 C6U3CK 10006134 IC50 = 1.8 nM T08856 CR7T3J 10009978 Ki = 672 nM T08856 C6DGR7 10027203 Ki = 1.3 nM T08856 CM52RO 10030422 IC50 = 0.77 nM T08856 CO39PK 10042482 Ki = 116 nM T08856 C19LUE 10050937 Ki = 32 nM T08856 CVTD42 10078499 Ki = 35000 nM T08856 CU7DJ1 10081163 Ki = 64000 nM T08856 C5W4ZA 10094362 IC50 = 10 nM T08856 C2XV5J 10098250 IC50 = 1.8 nM T08856 C0G7IY 10114318 Ki = 180 nM T08856 C78JHL 10116107 Ki = 260 nM T08856 C7OPQ8 10118047 IC50 = 140 nM T08856 C7A8MI 10120093 IC50 = 1.5 nM T08856 C7KR3Y 10136680 Ki = 220 nM T08856 CNU93J 10136924 Ki = 190 nM T08856 C1CDF2 10136925 Ki = 350 nM T08856 CJ9EX4 10138303 Ki = 60 nM T08856 CIH36M 10141214 IC50 = 170 nM T08856 CO6PS3 10162900 Ki = 210 nM T08856 CR5H6E 10163627 Ki = 1865 nM T08856 CZO5V4 10164317 IC50 = 0.5 nM T08856 CCX3T6 10183064 Ki > 15000 nM T08856 CK0P3F 10186536 Ki = 1957 nM T08856 CVRZ27 10198038 IC50 > 100000 nM T08856 CE1LI3 10204303 Ki = 200 nM T08856 CQFP69 10206106 Ki = 110 nM T08856 C4K1MJ 10208262 Ki > 3058 nM T08856 CV5X8A 10224181 IC50 > 100000 nM T08856 CGKU70 10224396 Ki = 220 nM T08856 C9CSG3 10226996 IC50 = 3100 nM T08856 C7T0WH 10229644 IC50 = 3 nM T08856 CQ1E4F 10248274 Ki = 7 nM T08856 CQJ0R3 10252900 Ki = 1.6 nM T08856 CGP97S 10274748 Ki = 730 nM T08856 C3IG0K 10280852 IC50 = 0.6 nM T08856 CDU36Y 10296475 Ki = 180 nM T08856 C48IRP 10296785 Ki = 150 nM T08856 C37ZDM 10317565 Ki = 270 nM T08856 CP1GW0 10318094 Ki = 0.3 nM T08856 CFQ4U0 10322451 Ki = 2 nM T08856 CY08WJ 10322755 Ki = 2050 nM T08856 C50KSE 10323483 IC50 = 10 nM T08856 CCZY62 10336856 IC50 = 20 nM T08856 C8C3AM 10337314 Ki = 489.78 nM T08856 CG6NT9 10338869 IC50 = 50 nM T08856 CJIW74 10343996 Ki < 2 nM T08856 C50DNH 10362338 Ki = 4 nM T08856 C9FU5G 10362663 IC50 = 1.5 nM T08856 CWIM61 10364088 IC50 = 14 nM T08856 CBA5I4 10365560 Ki = 0.7 nM T08856 C6T4WO 10370281 Ki = 13 nM T08856 CZNT94 10389113 IC50 = 15 nM T08856 CFKA79 10395015 Ki = 126 nM T08856 CA0TY8 10413076 Ki = 4 nM T08856 C98HMP 10413940 Ki = 9 nM T08856 C5WV1N 10439082 Ki = 428 nM T08856 C54UDR 10453826 IC50 = 200 nM T08856 CQUR30 10454592 Ki = 0.24 nM T08856 CP9WB1 10454818 Ki = 2 nM T08856 C6T8VC 10456675 Ki = 0.1 nM T08856 C8M9FE 10462640 Ki = 38900 nM T08856 CP30UC 10478059 Ki = 12 nM T08856 C87WDS 10478481 Ki < 1 nM T08856 C9VIP5 10479752 Ki = 30 nM T08856 CNQZ36 10483139 Ki = 170 nM T08856 CA7HT2 10498521 Ki = 20 nM T08856 C6KD0A 10498747 IC50 = 0.7 nM T08856 CL8O6I 10500340 Ki = 118 nM T08856 CGK80V 10500816 Ki = 39 nM T08856 CVID65 10500886 Ki = 21 nM T08856 C9YIS7 10501217 IC50 = 3 nM T08856 CP37WK 10501527 Ki = 19 nM T08856 C9DH4E 10501546 IC50 = 8 nM T08856 CK6YN5 10501862 Ki = 5 nM T08856 C9QE1B 10502327 Ki = 5 nM T08856 CZ1R5Q 10502869 Ki = 17 nM T08856 CO9S5H 10503708 Ki = 15 nM T08856 C86SGQ 10503952 Ki = 12000 nM T08856 CT2NM3 10505241 Ki = 17 nM T08856 C03MRW 10507152 Ki = 1 nM T08856 CC6H8T 10507755 Ki = 1.1 nM T08856 CXD8I5 10523292 Ki = 130 nM T08856 C90HBF 10523728 Ki = 10 nM T08856 CX6EB7 10524337 Ki = 390 nM T08856 CQTF46 10524338 Ki = 54 nM T08856 CYB53K 10525912 Ki = 43 nM T08856 C7HP4M 10527121 IC50 = 2 nM T08856 CZX87B 10529320 Ki = 9600 nM T08856 CGK37L 10529602 Ki = 2.4 nM T08856 CQ82VY 10530944 Ki = 28 nM T08856 CMJ23W 10540548 Ki = 50000 nM T08856 CB7P3Y 10544776 Ki = 194000 nM T08856 C0WHA9 10546565 Ki = 12 nM T08856 C40ZXE 10547784 Ki = 8 nM T08856 CAU9P2 10548378 IC50 = 100 nM T08856 CS10ZB 10549106 Ki = 8.5 nM T08856 C4PK0U 10549114 IC50 = 0.6 nM T08856 C5JS8L 10549329 Ki = 9 nM T08856 CG27UI 10549756 Ki = 45 nM T08856 C82HQE 10550145 Ki = 6 nM T08856 CWF2H8 10551771 IC50 = 70 nM T08856 C4K3UD 10552661 Ki = 16 nM T08856 CU8QP7 10552732 Ki = 11 nM T08856 C1ZHV9 10554637 IC50 = 8 nM T08856 CZ41HP 10554978 Ki = 21 nM T08856 C61BWV 10565981 Ki = 44000 nM T08856 CC8J5A 10566915 Ki = 1500 nM T08856 CIYR43 10570236 Ki = 41000 nM T08856 C6G3LP 10570582 IC50 = 30 nM T08856 CE14GM 10570702 IC50 = 10.6 nM T08856 CUQ29Z 10571396 Ki = 17 nM T08856 C42IAF 10573603 Ki = 13 nM T08856 CG39CF 10574279 Ki = 10 nM T08856 CT1OP7 10575767 IC50 = 2 nM T08856 CJ87EH 10576366 IC50 = 800 nM T08856 CVT1U6 10577196 IC50 = 500 nM T08856 CK05ZH 10579086 Ki = 1.2 nM T08856 C3R2SO 10580533 Ki = 2.5 nM T08856 CG87IY 10584303 Ki = 190000 nM T08856 CY09KX 10586834 Ki = 11000 nM T08856 C8J6HS 10591505 Ki = 123 nM T08856 C5VL8U 10592232 Ki = 9600 nM T08856 CB20LM 10594000 Ki = 31 nM T08856 CC69MB 10594682 IC50 = 20 nM T08856 CI71CK 10595804 Ki = 8 nM T08856 CD65NF 10597516 Ki = 29 nM T08856 CP2H8O 10597673 Ki = 7 nM T08856 C1W3FP 10600327 IC50 = 2 nM T08856 CN3E8J 10600844 Ki = 0.59 nM T08856 CEJ1U0 10603377 Ki = 32 nM T08856 C5G9MI 10610114 Ki = 1500 nM T08856 C06CAN 10619639 Ki = 13 nM T08856 CV14UH 10619971 Ki = 15 nM T08856 CSQ96T 10621933 Ki = 0.35 nM T08856 CVZ32G 10622447 Ki = 17 nM T08856 CU0JI9 10623424 IC50 = 2 nM T08856 CHRD92 10623565 Ki = 1400 nM T08856 C6R4EG 10624005 Ki = 1.2 nM T08856 C5FK4G 10624487 IC50 = 2000 nM T08856 CKF6D7 10625329 Ki = 5.2 nM T08856 C70MFZ 10626445 Ki = 23 nM T08856 C5VGB1 10626732 Ki = 30 nM T08856 CFBO63 10632558 Ki = 41000 nM T08856 CA63VQ 10640307 Ki = 35 nM T08856 C41RKE 10643401 Ki = 9 nM T08856 CUAI71 10643973 Ki = 1.5 nM T08856 CWEG60 10646580 IC50 = 3 nM T08856 CPYV83 10647658 Ki = 460 nM T08856 CD96LY 10648089 Ki = 0.56 nM T08856 CVX7Q2 10648390 Ki = 15 nM T08856 CT4IX1 10648424 IC50 = 3000 nM T08856 CC5B6L 10648524 Ki = 20000 nM T08856 C4TXZ1 10648776 Ki = 130 nM T08856 C07FPQ 10649518 Ki = 77 nM T08856 COT6B8 10650624 Ki = 34 nM T08856 C69SPO 10650906 Ki = 0.5 nM T08856 CT23XW 10650907 Ki = 1.4 nM T08856 C1U9GK 10658451 Ki = 2290.87 nM T08856 C3ELW7 10662922 Ki = 2290.87 nM T08856 C42SUO 10665403 Ki = 45000 nM T08856 C49AZV 10665669 IC50 = 4 nM T08856 CSCL07 10668823 Ki = 7.7 nM T08856 CFYC35 10669215 Ki = 3.3 nM T08856 C6TC0Z 10669216 Ki = 2.4 nM T08856 C4QVL0 10670896 Ki = 4 nM T08856 CGUT20 10671156 IC50 = 40 nM T08856 C3DXN5 10671411 Ki = 0.49 nM T08856 CWB19K 10671441 Ki = 1 nM T08856 CXDM24 10671863 Ki = 0.43 nM T08856 CNI5L7 10671934 IC50 = 200 nM T08856 CQT9E6 10672918 IC50 = 200 nM T08856 C8YB1A 10689487 Ki = 380 nM T08856 CU5M1J 10691797 Ki = 12 nM T08856 C8JX1G 10693698 Ki = 5 nM T08856 CM1T7K 10694510 Ki = 1.6 nM T08856 C7SM1E 10694604 Ki = 6.9 nM T08856 C7ZQM4 10695491 Ki = 0.29 nM T08856 CWS4N1 10695749 IC50 = 0.2 nM T08856 CN2UF8 10696122 IC50 = 800 nM T08856 CXL7E9 10696773 Ki = 4000 nM T08856 CG5JM9 10698412 Ki = 2 nM T08856 C56VSE 10698786 Ki = 1.3 nM T08856 C5E8QF 10707457 Ki = 125 nM T08856 CWYJ43 10717210 IC50 = 2 nM T08856 C0IL4Z 10717277 IC50 = 200 nM T08856 CES82X 10717319 IC50 = 80 nM T08856 C3TGW8 10717400 Ki = 108 nM T08856 CZ1M3L 10718058 Ki = 27 nM T08856 CQZ7M8 10718133 Ki = 21 nM T08856 CDNH67 10718890 IC50 = 20 nM T08856 CN8AK6 10718996 Ki = 0.11 nM T08856 C2IS9D 10719476 Ki = 0.49 nM T08856 CF46SQ 10721337 Ki = 27 nM T08856 CC1FB8 10721904 Ki = 2.1 nM T08856 CB2QD0 10723468 Ki = 1.3 nM T08856 CAL4W1 10728558 Ki = 52480.75 nM T08856 CO7VP4 10737552 Ki = 24 nM T08856 CB8G2D 10739728 Ki = 18 nM T08856 CJ6R1E 10740215 IC50 = 2 nM T08856 C4FWC9 10740485 Ki = 111 nM T08856 CQ9RW1 10740519 Ki = 1900 nM T08856 C0WKL7 10741470 Ki = 13 nM T08856 C0QT2F 10741956 Ki = 6 nM T08856 CY2BZ0 10742536 Ki = 58 nM T08856 C5BZ0J 10745489 Ki = 22 nM T08856 CK30AE 10745748 Ki = 1.5 nM T08856 CWF50D 10745851 Ki = 24 nM T08856 CA3F1N 10758013 Ki = 125 nM T08856 CHN73J 10759449 Ki = 300 nM T08856 CF7SH1 10761128 IC50 = 4 nM T08856 CDX13Z 10761730 Ki = 12 nM T08856 CA4U7D 10762262 Ki = 26 nM T08856 CP2G0N 10763745 Ki = 0.41 nM T08856 CFM5V2 10763804 IC50 = 8 nM T08856 CL0R4U 10764429 IC50 = 100 nM T08856 CM54WS 10764477 Ki = 531 nM T08856 C4ET3U 10764533 IC50 = 300 nM T08856 C4BY7G 10764534 IC50 = 30 nM T08856 CD58QP 10765874 IC50 = 100 nM T08856 CJW2B7 10766518 IC50 = 7 nM T08856 CA6C0Z 10766622 Ki = 0.6 nM T08856 C0R1ZA 10767025 Ki = 0.75 nM T08856 CNT4D0 10767387 Ki = 24 nM T08856 CAD6R8 10775444 Ki = 97723.72 nM T08856 CQ6U2Y 10780743 Ki = 24 nM T08856 C7TU1E 10783212 Ki = 8100 nM T08856 C15PVT 10785952 Ki = 24 nM T08856 CO19NM 10787883 Ki = 1600 nM T08856 C8AF9L 10787938 Ki = 0.34 nM T08856 C3P7LZ 10792025 Ki = 3.3 nM T08856 CY08PI 10792571 IC50 = 10 nM T08856 CG7VM1 10800736 Ki = 189000 nM T08856 CX5KJ0 10805200 Ki = 1900 nM T08856 C72ZQF 10807534 IC50 = 3000 nM T08856 CKV36G 10808884 IC50 = 3 nM T08856 C28WEN 10809988 Ki = 36000 nM T08856 CU9F7V 10810684 Ki = 27 nM T08856 C4UCQ8 10810983 IC50 = 50 nM T08856 CS0O7M 10811110 Ki = 21 nM T08856 C49VMO 10813119 IC50 = 3 nM T08856 CUOB87 10816515 Ki = 0.94 nM T08856 CO24DJ 10828912 Ki = 1100 nM T08856 CXI6S9 10832036 Ki = 2300 nM T08856 COE82D 10833334 Ki = 101 nM T08856 CJ8WG4 10833766 IC50 = 70 nM T08856 C9M1JI 10834357 Ki = 13 nM T08856 C3SZR1 10835069 IC50 = 2 nM T08856 CT3MN0 10837022 Ki = 6.5 nM T08856 CR0E9Q 10837740 Ki = 5.3 nM T08856 C9H4CP 10838922 Ki = 0.1 nM T08856 CR50UM 10839419 Ki = 7 nM T08856 CL1KG7 10840630 Ki = 31 nM T08856 CAIN04 10851204 Ki = 537.03 nM T08856 CAU0I3 10885834 IC50 = 3.631 nM T08856 CXHA75 10928874 IC50 = 2.692 nM T08856 C4JC9O 10930047 IC50 = 3.236 nM T08856 C7WEZ4 11009332 Ki = 36000 nM T08856 C9WPH7 11016072 Ki = 780 nM T08856 CBE68H 11016073 Ki = 4370 nM T08856 CG2DK0 11016448 IC50 = 1.5 nM T08856 CODQ51 11016616 IC50 = 1.5 nM T08856 CLXZ15 11037377 Ki = 0.45 nM T08856 C3W9IT 11046880 Ki = 70 nM T08856 C9RU4I 11059620 IC50 = 6.761 nM T08856 C1N5PT 11070986 IC50 = 5.3 nM T08856 C18EIZ 11071831 IC50 = 2.399 nM T08856 CR4V2D 11101785 Ki = 300 nM T08856 CY1SR9 11113744 IC50 = 25.8 nM T08856 C2YBQ7 11134935 IC50 = 3 nM T08856 CF52TX 11143173 Ki = 8600 nM T08856 C5WS3E 11147931 IC50 = 50000 nM T08856 CCQ6N8 11194666 IC50 = 40 nM T08856 CO76XI 11205873 IC50 = 30000 nM T08856 C9R7OM 11207122 IC50 = 90000 nM T08856 CUOH67 11252195 IC50 = 200 nM T08856 CP17ID 11284983 IC50 = 73 nM T08856 CF9O2R 11286824 IC50 > 100000 nM T08856 C1IW7N 11292680 IC50 = 1.6 nM T08856 C8C5AV 11294179 Ki > 10000 nM T08856 CLH50U 11318841 IC50 = 94 nM T08856 C0XR3B 11330861 IC50 = 110 nM T08856 CQH57S 11342435 IC50 = 42 nM T08856 CM8Y1J 11367571 IC50 = 10000 nM T08856 C13NCF 11400989 IC50 > 100000 nM T08856 CI0V6L 11447356 IC50 > 100000 nM T08856 COS67B 11456566 IC50 = 404 nM T08856 CCMT46 11457732 IC50 = 20000 nM T08856 CQ1D6E 11470070 IC50 = 80000 nM T08856 CJ46KN 11508259 Ki = 24 nM T08856 CCD93H 11730086 Ki = 480 nM T08856 C7CED0 11733417 IC50 = 294 nM T08856 CO8QT0 11753905 Ki = 2000 nM T08856 C1K6JY 11754185 IC50 = 1 nM T08856 C3P0TZ 11754739 Ki = 10 nM T08856 C5E7KU 11757592 Ki = 0.7 nM T08856 CSY8N7 11792237 IC50 = 1000 nM T08856 C7BV5P 11792968 Ki = 104 nM T08856 CX59YU 11792994 IC50 = 1000 nM T08856 CCSD72 11795621 IC50 = 2.4 nM T08856 CY8N1U 11795715 Ki = 4 nM T08856 CY7H2T 11795824 Ki = 10 nM T08856 CK24XT 11796481 Ki = 9 nM T08856 CWQ1S9 11797863 IC50 = 2 nM T08856 C37CLK 11798825 IC50 = 3 nM T08856 C3J4LX 11799180 Ki = 1700 nM T08856 C19RCP 11799753 Ki = 5.5 nM T08856 CQ9HE2 11811551 IC50 = 30.2 nM T08856 CLW3F1 11812791 IC50 = 44.67 nM T08856 C8DY3Z 11817193 IC50 = 4000 nM T08856 C02BWA 11967143 Ki = 272 nM T08856 CB80OT 12000718 IC50 = 3200 nM T08856 C43PJZ 12000720 IC50 > 20000 nM T08856 C0JID3 12447203 Ki > 100000 nM T08856 CTHQ39 12635073 Ki = 16000 nM T08856 CIQX87 12635074 Ki = 75000 nM T08856 C0XKJ1 12671872 IC50 = 70000 nM T08856 CQTX49 13738810 IC50 = 36000 nM T08856 C1AJO7 13968141 IC50 > 300000 nM T08856 CA2H8V 14303060 IC50 = 48 nM T08856 C1IZ7D 15296597 Ki = 19 nM T08856 CGH19T 15296844 IC50 > 300000 nM T08856 CK01NV 15379727 IC50 = 2 nM T08856 CV1HA9 15516783 IC50 = 36 nM T08856 CP2C4Z 15524387 Ki = 15300 nM T08856 CAF7R5 15524388 Ki = 9.2 nM T08856 C17HGN 15524389 Ki = 1192 nM T08856 CFH8Y6 15524390 Ki = 40000 nM T08856 C3N1KV 15629940 IC50 > 100000 nM T08856 C6R1LD 15985818 IC50 = 35 nM T08856 CS46XU 16126723 IC50 = 3.7 nM T08856 CYHI93 16418978 IC50 = 42900 nM T08856 CH7D2Q 16420684 IC50 = 6800 nM T08856 CQS0F5 16719301 IC50 > 10000 nM T08856 C75XDI 16730519 IC50 > 3000 nM T08856 C2W1VA 16739287 Ki = 200 nM T08856 CO21QH 18395616 IC50 = 19 nM T08856 C5B9WG 18533077 IC50 = 300 nM T08856 CS70KY 19366867 IC50 = 50 nM T08856 CIEH93 19382975 IC50 = 61000 nM T08856 CK8MP3 20620240 Ki = 80 nM T08856 CPC4G6 20620273 Ki = 260 nM T08856 C26UJT 20620561 IC50 = 120 nM T08856 C2E3CY 20620614 IC50 = 190 nM T08856 CVEX54 20620688 IC50 = 67 nM T08856 CV1SD8 20620714 IC50 = 6.7 nM T08856 C3GAC4 20620715 IC50 = 49 nM T08856 C7QV8K 20620757 IC50 = 1100 nM T08856 CVO73Y 20620827 IC50 = 1200 nM T08856 CQ14NY 20620831 IC50 = 700 nM T08856 C5RQ8A 20620860 IC50 = 100 nM T08856 CA7FK0 20639531 IC50 = 15 nM T08856 CMX23W 20639537 IC50 = 14 nM T08856 C34XRP 20639540 IC50 = 25 nM T08856 C7AP8Z 20639546 IC50 = 125 nM T08856 CPK09X 20651316 IC50 = 0.7 nM T08856 C4I1OM 20735209 IC50 = 10000 nM T08856 CE5DH1 22484408 IC50 = 2.6 nM T08856 CZT05X 22484417 Ki = 900 nM T08856 CZT64B 22484431 Ki = 180 nM T08856 CAM10T 22485252 IC50 = 30 nM T08856 CAY3N6 22485292 IC50 = 1.8 nM T08856 C3YL5X 22485311 IC50 = 1.6 nM T08856 CWA03L 22485327 IC50 = 1.9 nM T08856 C5JZF1 22485344 IC50 = 4 nM T08856 CI7MY5 22485346 IC50 = 2.4 nM T08856 CI1YL7 22485347 IC50 = 1.2 nM T08856 C25OBD 22485356 IC50 = 1.8 nM T08856 CL64TJ 22485368 IC50 = 1.4 nM T08856 CT4GF9 22485381 IC50 = 9400 nM T08856 C27NDB 22485386 IC50 = 2 nM T08856 C3MG9P 22485396 IC50 = 2.4 nM T08856 CZY10U 22485408 IC50 = 1.4 nM T08856 C89AGT 22485413 IC50 = 1.3 nM T08856 C03NLM 22485417 IC50 = 0.4 nM T08856 C8GHU9 22485432 IC50 = 1.5 nM T08856 CWPM36 22642543 IC50 = 1 nM T08856 C5EQ7I 22642544 IC50 = 8 nM T08856 CD71UM 22642553 IC50 = 2 nM T08856 CRL2G4 22642563 IC50 = 3 nM T08856 C2Q4XK 22707806 IC50 = 1.6 nM T08856 CIYA45 22985930 IC50 = 0.7 nM T08856 C9GKH3 23523881 IC50 = 3 nM T08856 CU8O7L 23523890 IC50 = 8 nM T08856 CSXG85 23523891 IC50 = 2 nM T08856 CV85UI 23523893 IC50 = 200 nM T08856 CXZ20T 23523894 IC50 = 20 nM T08856 CPLS94 23523896 IC50 = 3000 nM T08856 CM0K4X 23523897 IC50 = 10 nM T08856 CBI65T 23523899 IC50 = 200 nM T08856 CP6ZF2 23523900 IC50 = 20 nM T08856 CGWL84 23523905 IC50 = 800 nM T08856 CY7RC8 23523909 IC50 = 2 nM T08856 CV06HF 23523910 IC50 = 300 nM T08856 CU8BN9 23523911 IC50 = 30 nM T08856 C5GR7Y 23523914 IC50 = 100 nM T08856 CD3U8A 23627203 Ki = 2700 nM T08856 C8UIC6 23644662 Ki > 100000 nM T08856 CCLA40 23644663 Ki > 100000 nM T08856 CSZ6J4 23645528 Ki = 4.9 nM T08856 C6UH9Q 23645529 Ki = 1.1 nM T08856 CD0JP3 23645530 Ki = 1 nM T08856 CM37EC 23645531 Ki = 4.2 nM T08856 C9PD5F 23645532 Ki = 5.1 nM T08856 C1OE7R 23645533 Ki = 1.1 nM T08856 CCSN04 23645534 Ki = 2.3 nM T08856 CU08WI 23645535 Ki = 0.3 nM T08856 CY41UC 23645536 Ki = 18 nM T08856 CX15EH 23645537 Ki = 6.4 nM T08856 CD3Q6G 23645538 Ki = 27 nM T08856 CE6NQ2 23645539 Ki = 25000 nM T08856 C4VK3U 23645540 Ki = 23000 nM T08856 C8VM1C 23645541 Ki = 76000 nM T08856 C0MUT6 23645542 Ki = 15000 nM T08856 CNI07H 23645543 Ki = 16000 nM T08856 CHK2X1 23645544 Ki = 24000 nM T08856 CW1V2Z 23645545 Ki = 16000 nM T08856 C6SP7T 23645546 Ki = 10000 nM T08856 CD9QO2 23645547 Ki = 1000 nM T08856 C25YLZ 23645548 Ki = 120 nM T08856 COIZ43 23655713 IC50 = 754 nM T08856 CURM98 23655714 IC50 = 71000 nM T08856 CO90JC 23655717 IC50 = 2460 nM T08856 C56NMQ 23655910 IC50 = 7480 nM T08856 C9QZX5 23655911 IC50 = 6760 nM T08856 CA8W3K 23656106 IC50 = 12 nM T08856 CU4R7T 23656291 IC50 = 2 nM T08856 CVZ2M1 23656293 IC50 = 3 nM T08856 CL5C1I 23656295 IC50 = 75 nM T08856 CZP12E 23656450 IC50 = 20 nM T08856 CA2PY5 23657418 IC50 = 105 nM T08856 CN9TY1 23657419 IC50 = 1200 nM T08856 C9FHZ1 23657421 IC50 = 18 nM T08856 CY9LF1 23657422 IC50 = 0.9 nM T08856 C28SPW 23657691 IC50 = 14000 nM T08856 CVJ1T7 23657695 IC50 = 78000 nM T08856 CAL05Q 23657697 IC50 = 22000 nM T08856 CAG3Q8 23667877 IC50 = 40 nM T08856 C6AW7U 23692637 IC50 > 100000 nM T08856 C3TWS6 24178109 Ki = 4.6 nM T08856 C35QME 24742028 IC50 = 2 nM T08856 C18FRG 24807817 IC50 = 50000 nM T08856 CNR3U7 24866945 IC50 = 25500 nM T08856 CFL04M 24881245 IC50 = 150000 nM T08856 CLIC14 24881246 IC50 = 70000 nM T08856 CAQ9Z1 25022681 Ki > 3058 nM T08856 CA86UE 25049752 Ki = 9 nM T08856 C82NLV 25049754 Ki = 173 nM T08856 C6QFV4 25049756 Ki = 240 nM T08856 CX6D9J 25138245 Ki = 90 nM T08856 C7A6JQ 25138250 Ki = 200 nM T08856 CR35QP 25144971 IC50 = 57 nM T08856 C0Y5BC 25145683 IC50 = 7.4 nM T08856 CB7V8Y 25147773 IC50 = 0.29 nM T08856 C3KF1V 25178145 IC50 = 0.74 nM T08856 CG5Y2R 25178357 IC50 = 4.3 nM T08856 C4PZY6 25180866 IC50 = 29.2 nM T08856 CEP9Q2 25180867 IC50 = 0.4 nM T08856 C9HZG2 25181078 IC50 = 8200 nM T08856 CMYP34 25181079 IC50 = 4360 nM T08856 C7U1YC 25181080 IC50 = 59 nM T08856 C85HLG 25181081 IC50 = 35 nM T08856 CHR2P1 25183768 Ki > 25000 nM T08856 CT80ED 44219901 IC50 = 1700 nM T08856 C94JVY 44219902 IC50 = 3600 nM T08856 C7J6GH 44219903 IC50 = 66 nM T08856 C9J7WL 44219904 IC50 = 7600 nM T08856 CRQ71E 44219905 IC50 = 440 nM T08856 C4Z0ID 44219906 IC50 = 140 nM T08856 CRNA25 44220092 IC50 = 110 nM T08856 C9T5ZF 44220093 IC50 = 63 nM T08856 CV38TE 44222825 IC50 = 560 nM T08856 CJI73R 44222826 IC50 = 37 nM T08856 CGQ30N 44222827 IC50 = 65 nM T08856 CCI64J 44224245 IC50 = 37 nM T08856 CLRT69 44247751 IC50 = 5.1 nM T08856 CAR34Y 44263877 IC50 = 47.3 nM T08856 CEV08N 44263913 IC50 = 3.3 nM T08856 C5ZI0X 44263926 IC50 = 1.5 nM T08856 CO3C1E 44263994 IC50 = 6.6 nM T08856 C9XJ7U 44264020 IC50 = 102 nM T08856 C6L0MJ 44264021 IC50 = 3.7 nM T08856 CJ1WE7 44264036 IC50 = 2.8 nM T08856 C50QFR 44264375 IC50 = 6.3 nM T08856 C6YT3K 44280285 Ki = 102 nM T08856 CC2O3U 44280323 Ki = 4 nM T08856 CIE09F 44280336 Ki = 0.5 nM T08856 CI9L2E 44280411 Ki = 163 nM T08856 CC2QR7 44281720 Ki = 7 nM T08856 CN23FC 44282968 IC50 = 3000 nM T08856 C2TV5I 44282969 IC50 = 80 nM T08856 CG3LF0 44282970 IC50 = 300 nM T08856 CZ2AL1 44286483 IC50 > 120000 nM T08856 C5XS0I 44294322 Ki = 293 nM T08856 CI75VF 44299758 IC50 = 5 nM T08856 CTF47Y 44299811 IC50 = 20 nM T08856 CS1Q3J 44299812 IC50 = 30 nM T08856 CY8XI5 44299813 IC50 = 500 nM T08856 CCS1I4 44299817 IC50 = 7 nM T08856 CKU1O9 44299818 IC50 = 2000 nM T08856 C3EB9S 44299821 IC50 = 300 nM T08856 C6CLM4 44299832 IC50 = 30 nM T08856 CT1ZQ8 44299853 IC50 = 9 nM T08856 CFR75V 44299935 IC50 = 2 nM T08856 C17ENS 44299950 IC50 = 10 nM T08856 CLF24Y 44299978 IC50 = 600 nM T08856 CJI38H 44299979 IC50 = 20 nM T08856 CE7DN4 44299980 IC50 = 40 nM T08856 CM3FT6 44299984 IC50 = 90 nM T08856 CC2X8J 44299988 IC50 = 2 nM T08856 C4JI5K 44299989 IC50 = 5 nM T08856 CCNK46 44299992 IC50 = 10 nM T08856 C35WLI 44299996 IC50 = 300 nM T08856 CX06GL 44299999 IC50 = 30 nM T08856 C3SJL1 44300006 IC50 = 60 nM T08856 C6PMI7 44300007 IC50 = 20 nM T08856 C87BFW 44300015 IC50 = 20 nM T08856 C86OPX 44300033 IC50 = 10 nM T08856 C3CP7G 44300047 IC50 = 3000 nM T08856 CNS97M 44300048 IC50 = 20 nM T08856 CO59XG 44300051 IC50 = 40 nM T08856 CP31DY 44300057 IC50 = 200 nM T08856 CEFB86 44300058 IC50 = 1000 nM T08856 CISL43 44300063 IC50 = 7000 nM T08856 CWHX49 44300103 IC50 = 2000 nM T08856 C5M1VZ 44300163 IC50 = 10 nM T08856 CN73OS 44300183 IC50 = 80 nM T08856 COW30X 44300184 IC50 = 4000 nM T08856 C4PNM3 44300199 IC50 = 80 nM T08856 C5R7AL 44300210 IC50 = 30 nM T08856 CZN37U 44300222 IC50 = 600 nM T08856 C5VY0B 44300223 IC50 = 10 nM T08856 CI13FM 44300231 IC50 = 20 nM T08856 CP7M0F 44300252 IC50 = 90 nM T08856 CZUY51 44310789 Ki = 4.5 nM T08856 CH92OI 44310813 Ki = 4.5 nM T08856 CI4Y5N 44310825 Ki = 14 nM T08856 C5W8QH 44310847 Ki = 3.7 nM T08856 CLQV12 44310863 Ki = 0.45 nM T08856 CR70EA 44310887 Ki = 0.66 nM T08856 CJ9T1F 44310904 Ki = 0.96 nM T08856 CN9P5A 44310921 Ki = 0.64 nM T08856 CXB76U 44310932 Ki = 1.3 nM T08856 CMW5G3 44310933 Ki = 13 nM T08856 CBY0T1 44310973 Ki = 13 nM T08856 C5D9FS 44311011 Ki = 0.3 nM T08856 C95RKF 44311052 Ki = 3.6 nM T08856 C2GC9W 44311172 Ki = 7.7 nM T08856 C0K1IL 44311187 Ki = 0.54 nM T08856 CL3CS0 44311254 Ki = 7.8 nM T08856 CV63JP 44311265 Ki = 0.7 nM T08856 CS56ER 44311267 Ki = 73 nM T08856 C5MBT7 44311268 Ki = 6.2 nM T08856 CM64HK 44311313 Ki = 0.33 nM T08856 CU5X4G 44311331 Ki = 0.63 nM T08856 CLQ48B 44311332 Ki = 6.8 nM T08856 C5AO7Z 44311335 Ki = 0.82 nM T08856 C78TEU 44311349 Ki = 1.7 nM T08856 CJEM64 44311491 Ki = 0.65 nM T08856 C2W5NQ 44311510 Ki = 0.53 nM T08856 C2MIT8 44311525 Ki = 1 nM T08856 CP7L6Q 44311566 Ki = 2.4 nM T08856 C0B4HZ 44312333 Ki = 20 nM T08856 CH48TD 44315155 IC50 = 12 nM T08856 C62FXJ 44315244 IC50 = 0.56 nM T08856 C50IQE 44315333 IC50 = 2.1 nM T08856 CG0JD3 44316269 Ki = 13000 nM T08856 C1O6PM 44316416 Ki = 9 nM T08856 CP83EX 44316470 Ki = 7000 nM T08856 CLOS38 44316842 Ki = 6 nM T08856 C89IQW 44318090 IC50 = 3.2 nM T08856 CJU31O 44321285 Ki = 4.5 nM T08856 C41VFA 44321286 Ki = 2.5 nM T08856 C5S2ZU 44321484 Ki = 20 nM T08856 CLQ23M 44321485 Ki = 40 nM T08856 CHF76Q 44321540 Ki = 4 nM T08856 CVOL49 44321593 Ki = 7.5 nM T08856 CB97GK 44321601 Ki = 3.5 nM T08856 CT0O7Y 44321602 Ki = 25 nM T08856 CU62BP 44321746 Ki = 5.5 nM T08856 CQU2K9 44321782 Ki = 17 nM T08856 CV8T3N 44321783 Ki = 5 nM T08856 CIBO50 44321801 Ki = 0.7 nM T08856 C4E8GU 44321802 Ki = 34 nM T08856 CYDN18 44321803 Ki = 7 nM T08856 C7Z4DQ 44321887 Ki = 5 nM T08856 CFJ20T 44321932 Ki = 1.5 nM T08856 C9O0VB 44321965 Ki = 240 nM T08856 C2E3RF 44321966 Ki = 6 nM T08856 CW9S1N 44321967 Ki = 230 nM T08856 C1FI3O 44321975 Ki < 0.5 nM T08856 CLB8J6 44321976 Ki = 20 nM T08856 CR0KN1 44322209 Ki = 240 nM T08856 C5LE1P 44322210 Ki = 8 nM T08856 CQ7AW8 44322211 Ki = 19 nM T08856 CJY2O7 44322214 Ki = 45 nM T08856 CR9GI0 44322215 Ki = 4.3 nM T08856 C7V5EF 44326167 IC50 = 20 nM T08856 C93HSL 44326184 IC50 = 70 nM T08856 CY3I9B 44326185 IC50 = 3 nM T08856 C23OQF 44326225 IC50 = 30 nM T08856 CY3GH5 44326232 IC50 = 15 nM T08856 C6E9IV 44326443 IC50 = 80 nM T08856 C85QTP 44328155 IC50 > 100000 nM T08856 CZQ6N7 44328189 IC50 = 30000 nM T08856 C90CHA 44329405 IC50 = 100 nM T08856 C2PB4Z 44329622 IC50 = 1000 nM T08856 CI3Z4K 44329623 IC50 = 10 nM T08856 C6OL8M 44329636 IC50 = 100 nM T08856 CB0G1H 44329644 IC50 = 3981.07 nM T08856 CA65RO 44329672 IC50 = 100 nM T08856 CK9HO7 44329673 IC50 = 600 nM T08856 C07GRS 44329693 IC50 = 3 nM T08856 CBH16R 44329694 IC50 = 10 nM T08856 CG3E7A 44329712 IC50 = 2 nM T08856 C9SN6I 44329713 IC50 = 90 nM T08856 CZ2FW6 44329725 IC50 = 39.81 nM T08856 CDKI48 44329741 IC50 = 10 nM T08856 CK3M2H 44329742 IC50 = 199.53 nM T08856 C39RDS 44329886 IC50 = 3.981 nM T08856 C63RHP 44329909 IC50 = 3.02 nM T08856 CVQA75 44329910 IC50 = 19.95 nM T08856 C84SLI 44329926 IC50 = 4 nM T08856 CJS6B1 44329927 IC50 = 9 nM T08856 C1IE0S 44330147 IC50 > 100000 nM T08856 CL9I4M 44341538 Ki = 303 nM T08856 CE3MT4 44341611 Ki = 18400 nM T08856 CJTZ45 44341652 Ki = 200000 nM T08856 C2SZB1 44342614 IC50 = 2 nM T08856 CVZH63 44343240 Ki = 55000 nM T08856 CG7B9Y 44343258 Ki = 50000 nM T08856 CY54GC 44343397 Ki = 168000 nM T08856 C65API 44343404 Ki = 88000 nM T08856 C1JS3R 44343507 Ki = 35000 nM T08856 CQ76PY 44343526 Ki = 26000 nM T08856 CU6ZK2 44343534 Ki = 25000 nM T08856 C8G7WL 44344564 Ki = 190 nM T08856 CD43AB 44344565 Ki = 100 nM T08856 CC29QO 44344739 Ki = 170 nM T08856 CWA42F 44344746 Ki = 4.7 nM T08856 CQPN17 44344749 Ki < 2 nM T08856 CL41FG 44344753 Ki = 4200 nM T08856 C1LE9J 44359497 IC50 = 800 nM T08856 CHE08D 44359498 IC50 = 7000 nM T08856 C4Z5RV 44359507 IC50 = 3 nM T08856 C2HZ6K 44359536 IC50 = 80 nM T08856 C1J4KA 44359537 IC50 = 200 nM T08856 CV4ZM1 44359563 IC50 = 8 nM T08856 CP1CD9 44359641 IC50 = 2 nM T08856 CI5FY8 44359659 IC50 = 2 nM T08856 CJB74Y 44359661 IC50 = 5 nM T08856 CC9LH6 44359662 IC50 = 500 nM T08856 CHW43J 44359663 IC50 = 20 nM T08856 C17QMW 44359665 IC50 = 3000 nM T08856 CKD2L0 44359666 IC50 = 20 nM T08856 CJ2QU8 44359668 IC50 = 40 nM T08856 CKM4W6 44359670 IC50 = 2000 nM T08856 CC7UB0 44359671 IC50 = 30 nM T08856 CJ91ZQ 44359676 IC50 = 2000 nM T08856 CY4CA6 44359677 IC50 = 10 nM T08856 C92OKL 44359678 IC50 = 1 nM T08856 CHWK87 44359686 IC50 = 500 nM T08856 CEDO94 44359692 IC50 = 2 nM T08856 CC96HP 44359693 IC50 = 100 nM T08856 CHZK92 44359695 IC50 = 1000 nM T08856 C6XBP4 44359701 IC50 = 30 nM T08856 C2C7LJ 44359712 IC50 = 2 nM T08856 CVA09S 44359714 IC50 = 3000 nM T08856 CNX27J 44359717 IC50 = 70 nM T08856 CLG0O4 44359719 IC50 = 10 nM T08856 CZL92R 44359720 IC50 = 300 nM T08856 C3T0BS 44359739 IC50 = 90 nM T08856 CCN30T 44359740 IC50 = 30 nM T08856 C3NIL4 44359744 IC50 = 90 nM T08856 CR7E8B 44359745 IC50 = 20 nM T08856 CP02BN 44359746 IC50 = 60 nM T08856 CX65KF 44359747 IC50 = 2 nM T08856 C8PKH7 44359748 IC50 = 30 nM T08856 CJ41AC 44359758 IC50 = 2000 nM T08856 CNSL71 44359759 IC50 = 40 nM T08856 CZ4E9Q 44359760 IC50 = 50 nM T08856 C7NTP1 44359790 IC50 = 80 nM T08856 CHXE26 44359791 IC50 = 80 nM T08856 C7VI5F 44359792 IC50 = 40 nM T08856 CAI78D 44359808 IC50 = 300 nM T08856 CN0BH2 44359811 IC50 = 9 nM T08856 CYL4P0 44359813 IC50 = 2 nM T08856 CO7LW8 44359868 IC50 = 20 nM T08856 CAK2S0 44359869 IC50 = 40 nM T08856 CX9J2G 44359888 IC50 = 2 nM T08856 CU9I5B 44359889 IC50 = 600 nM T08856 CLZG86 44359923 IC50 = 10 nM T08856 CF0P9S 44359924 IC50 = 200 nM T08856 CIL92Y 44359925 IC50 = 7 nM T08856 CR35WH 44359926 IC50 = 20 nM T08856 CK6MD8 44360002 IC50 = 30 nM T08856 CL4F1H 44360016 IC50 = 20 nM T08856 CRW61Q 44360082 IC50 = 10 nM T08856 C9XZQ3 44360104 IC50 = 10 nM T08856 C4PF0M 44360162 IC50 = 600 nM T08856 C3IW9L 44360784 IC50 = 1.9 nM T08856 CV0T6G 44383797 Ki = 7000 nM T08856 C9NIT7 44383842 Ki = 14000 nM T08856 CDQV80 44384020 Ki = 300 nM T08856 CA2L3U 44384021 Ki = 28000 nM T08856 CT1MN8 44384090 Ki = 6000 nM T08856 C8OKQ9 44384146 Ki = 75000 nM T08856 C5C3LY 44384231 Ki = 1000 nM T08856 CILQ34 44384272 Ki = 38000 nM T08856 CIJ61R 44384273 Ki = 430 nM T08856 CQ2UE9 44384356 Ki = 1500 nM T08856 C14RMP 44384416 Ki = 1000 nM T08856 C5MO9Q 44384474 Ki = 3000 nM T08856 CUMQ67 44384980 Ki = 250 nM T08856 C3CG5I 44385039 Ki = 22000 nM T08856 CE7V9A 44385250 Ki = 6000 nM T08856 CE5RJ0 44385333 Ki = 1700 nM T08856 CNPO26 44390575 IC50 = 10 nM T08856 CC7QW9 44391352 IC50 = 31 nM T08856 CZB81D 44395506 IC50 = 1 nM T08856 CWGQ46 44404503 IC50 = 52 nM T08856 CLXM58 44404504 IC50 = 101 nM T08856 C0G4MR 44405997 IC50 > 380000 nM T08856 CZ0XC1 44405998 IC50 = 1000000 nM T08856 C1F0DR 44406571 IC50 = 10 nM T08856 CHM26J 44406652 Ki = 17 nM T08856 C1K3QM 44406655 IC50 = 20 nM T08856 CT5PC9 44422672 IC50 = 0.39 nM T08856 CS9D5U 44422720 IC50 = 0.37 nM T08856 CNWM05 44422723 IC50 = 1.5 nM T08856 C58LAY 44422724 IC50 = 1.1 nM T08856 CDQU41 44422736 IC50 = 2.4 nM T08856 CVUB56 44422737 IC50 = 1.3 nM T08856 CB8G2W 44422743 IC50 = 0.4 nM T08856 CFX42T 44422744 IC50 = 260 nM T08856 C9EL7F 44422749 IC50 = 110 nM T08856 CWU7G8 44434565 IC50 = 101 nM T08856 C1YT3E 44445914 Ki = 190546.07 nM T08856 CG0Z7I 44478924 IC50 = 1900 nM T08856 CFO27Y 44478926 IC50 = 280 nM T08856 CBZJ29 44478927 IC50 = 120 nM T08856 CRJ24K 44479197 IC50 = 54 nM T08856 CGOH82 44479198 IC50 = 1200 nM T08856 CLV56M 44479199 IC50 = 99 nM T08856 CY92OQ 44479458 IC50 = 9200 nM T08856 CH1QG9 44479459 IC50 = 87 nM T08856 CB1NT7 44479460 IC50 = 370 nM T08856 C0JQ9L 44479699 IC50 = 390 nM T08856 C0DN1Q 44479700 IC50 = 74000 nM T08856 CTG24W 44479702 IC50 = 1900 nM T08856 CGZ49M 44479703 IC50 = 290 nM T08856 CAK94X 44563337 IC50 = 1010 nM T08856 CK68GT 44580539 Ki = 3.01 nM T08856 CACH13 45269631 IC50 = 48 nM T08856 CMPE63 45482676 IC50 = 2000 nM T08856 CL2U4Z 46829322 Ki = 13 nM T08856 C5L8GF 46871738 IC50 = 670 nM T08856 CR1KF7 46871739 IC50 = 1000 nM T08856 C8Q6YR 46871740 IC50 = 59.2 nM T08856 C58YSM 46871741 IC50 > 10000 nM T08856 C0YR7M 46938728 IC50 = 0.4 nM T08856 C2S7PK 46942365 Ki = 9.1 nM T08856 C7XW1Q 50907084 Ki = 8 nM T08856 C8RL5Q 50907292 Ki = 48 nM T08856 CU2SX3 51355576 Ki > 10000 nM T08856 CLA96C 53232689 Ki = 250 nM T08856 CZ06OY 53233469 IC50 = 140 nM T08856 CWH47R 53319228 Ki = 10 nM T08856 C4UE6R 53322469 IC50 > 100000 nM T08856 CPY02U 53327890 IC50 = 490 nM T08856 CPGE80 53327891 IC50 = 280 nM T08856 CLJ4G2 53328858 IC50 = 200 nM T08856 C4G3QL 53328859 IC50 = 500 nM T08856 CX1TW0 53328860 IC50 = 30 nM T08856 C0ZX5G 53329215 IC50 = 440 nM T08856 CSU52A 53329216 IC50 = 1700 nM T08856 C6Y2EV 53374826 IC50 > 100000 nM T08856 C3LF0P 54580544 Ki = 140 nM T08856 CA8U9V 54580837 IC50 > 10000 nM T08856 CVO09J 54581546 Ki = 240 nM T08856 CWB2Q6 54581896 IC50 = 800 nM T08856 CD09BZ 54582543 IC50 = 1200 nM T08856 CK52YD 54583511 Ki = 74 nM T08856 CF0SK8 54583712 IC50 = 31 nM T08856 CG37UX 54587429 Ki = 72 nM T08856 C71KLJ 54679182 IC50 = 21900 nM T08856 C62FZC 56835063 IC50 = 154 nM T08856 CKJ9S1 56835167 IC50 = 21 nM T08856 C21CLZ 56835168 IC50 = 67 nM T08856 C0L2TS 56835169 IC50 = 300 nM T08856 C8TH2F 56945850 IC50 = 129 nM T08856 CD72TG 56945851 IC50 = 15 nM T08856 C8J4SC 56945854 IC50 = 48 nM T08856 C1AIZ6 56945963 IC50 = 49 nM T08856 CXQC91 56945964 IC50 = 58 nM T08856 CM4H9D 56945965 IC50 = 150 nM T08856 CUT4S2 56946063 IC50 = 107 nM T08856 C2CQR8 56946064 IC50 = 27 nM T08856 C2H8PG 56946065 IC50 = 19 nM T08856 CW2P6A 56946167 IC50 = 15 nM T08856 CT8S3G 56946168 IC50 = 116 nM T08856 CQU16V 57339411 Ki = 75 nM T08856 C6LM3B 57339412 Ki = 43 nM T08856 CNVG85 57339413 Ki = 14 nM T08856 C0KPD8 57384084 IC50 = 400 nM T08856 CV67JB 57384091 IC50 = 100 nM T08856 C0G2VY 57403564 IC50 = 4 nM T08856 C2MH8O 57523473 IC50 = 0.11 nM T08856 C57CEM 57523505 IC50 = 3 nM T08856 CS8W4L 57523538 IC50 = 14 nM T08856 CIT7B9 57523539 IC50 = 0.2 nM T08856 C56QXU 57523540 IC50 = 5 nM T08856 CX8IU3 57523541 IC50 = 58 nM T08856 CE8CL9 57523575 IC50 = 8 nM T08856 CWUP89 57523576 IC50 = 0.02 nM T08856 CT2QS3 57523577 IC50 = 0.03 nM T08856 CK6M0Y 57523578 IC50 = 0.04 nM T08856 C0HVU7 57523611 IC50 = 5 nM T08856 C5Q0ND 57523641 IC50 = 9 nM T08856 C1PHI6 57708731 IC50 > 1000 nM T08856 CF2Z7W 57708783 IC50 = 21 nM T08856 C9KV2W 57708792 IC50 = 110 nM T08856 CE36GP 57708799 IC50 = 76 nM T08856 C23QGY 57708843 IC50 = 480 nM T08856 C2J5CW 57708880 IC50 = 510 nM T08856 C1K6AP 57708886 IC50 = 11 nM T08856 CY1N3J 57792153 IC50 = 1010 nM T08856 C1EJ4S 59379730 Ki = 0.71 nM T08856 CAT67H 59910477 IC50 = 56.2 nM T08856 CFM0Q5 70690777 IC50 = 0.5 nM T08856 CY4E9Z 70692916 IC50 > 100000 nM T08856 COM1B0 71449369 IC50 = 715 nM T08856 CA7M9F 71451166 IC50 = 8200 nM T08856 CD4CP2 71451167 IC50 = 4500 nM T08856 C6M9VL 71451168 IC50 = 2600 nM T08856 C7HUF5 71451169 IC50 = 313 nM T08856 CMW3O0 71451330 Ki > 200000 nM T08856 CE98YL 71452999 IC50 = 266 nM T08856 C8VC6N 71453000 IC50 = 109 nM T08856 C4VKI1 71453001 IC50 = 586 nM T08856 CGCM02 71454432 IC50 = 3000 nM T08856 C7U2RT 71454740 IC50 = 63000 nM T08856 C9QS6E 71456659 Ki = 2.5 nM T08856 CXC1U7 71458350 IC50 = 184 nM T08856 C4IZ5V 71458351 IC50 = 153 nM T08856 CZO86D 71460193 IC50 = 271 nM T08856 CWL97M 71461905 IC50 = 336 nM T08856 CUT3H5 71461906 IC50 = 210 nM T08856 C06AXC 71461907 IC50 = 66 nM T08856 CSW59Y 71461908 IC50 = 2020 nM T08856 C3L7SD 71533484 IC50 = 217 nM T08856 CZH5S9 71533485 IC50 = 282 nM T08856 CGM72Q 71540498 IC50 = 44 nM T08856 CXA1I5 71540599 IC50 = 85 nM T08856 C7CV9E 71540600 IC50 = 60 nM T08856 CA4BP6 71540601 IC50 = 117 nM T08856 CMZ3T2 71540715 IC50 = 88 nM T08856 CXY83G 71540716 IC50 = 98 nM T08856 C1ZH2G 71540717 IC50 = 91 nM T08856 CT4UD5 71540831 IC50 = 125 nM T08856 CP7SX8 71540832 IC50 = 162 nM T08856 C9IW7R 71540833 IC50 = 46 nM T08856 CKV2U5 71817094 Ki = 32 nM T08856 CHDS52 71817095 Ki = 98 nM T08856 C5LZH0 71817097 Ki = 3 nM T08856 C50SID 71817098 Ki = 20 nM T08856 CN83DB 71817100 Ki = 37 nM T08856 CX4G0R 72204928 IC50 > 100000 nM T08856 CG9C6U 72204929 IC50 = 2400 nM T08856 C5A6XZ 72204930 IC50 = 15000 nM T08856 C0XZK4 72204931 IC50 > 100000 nM T08856 CM8Y7X 72204932 IC50 > 100000 nM T08856 C6RY4X 72204933 IC50 > 100000 nM T08856 C4N5AB 72204934 IC50 > 100000 nM T08856 C3H2FZ 72205111 IC50 > 100000 nM T08856 CQ0VX7 72205112 IC50 > 100000 nM T08856 CQ7TI1 72205113 IC50 = 44000 nM T08856 CPAW52 72205114 IC50 = 39900 nM T08856 C2LD3J 72205115 IC50 = 43000 nM T08856 CE4J8F 72711063 Ki = 15000 nM T08856 CC0ZX4 72714092 Ki = 11000 nM T08856 CE51LQ 72714333 Ki = 15000 nM T08856 CH4VF7 72714336 Ki = 17000 nM T08856 C9FL7V 72714339 Ki = 13000 nM T08856 CDX2F9 72984326 IC50 = 2.97 nM T08856 CUKG79 73292708 IC50 = 2 nM T08856 C5D3CJ 73292709 IC50 = 1 nM T08856 CL69NM 73292710 IC50 = 1 nM T08856 CQ4RO1 73292711 IC50 = 0.4 nM T08856 C7CT2E 73292869 IC50 = 1 nM T08856 CA0LS6 73292870 IC50 = 0.5 nM T08856 CJU3V6 73292871 IC50 = 0.2 nM T08856 C3PGF2 73292872 IC50 = 1 nM T08856 C0O8VM 73292873 IC50 = 0.9 nM T08856 CBR9I5 73293034 IC50 = 2 nM T08856 C9FD2C 73293035 IC50 = 4 nM T08856 C7LP5J 73293036 IC50 = 0.4 nM T08856 C9PQG1 73293037 IC50 = 35 nM T08856 C4PF1H 73293038 IC50 = 0.05 nM T08856 CE39WF 73293196 IC50 = 0.7 nM T08856 CU96XE 73293197 IC50 = 5 nM T08856 CGC51Z 73293198 IC50 = 2 nM T08856 CC83FW 73293199 IC50 = 0.2 nM T08856 CS6T8M 73293200 IC50 = 0.3 nM T08856 CW5IQ0 73345859 Ki = 6 nM T08856 C25SOB 73349251 IC50 = 0.3 nM T08856 CW01EA 73349535 IC50 = 47000 nM T08856 C43WKX 73353429 Ki = 4 nM T08856 CK42DO 73353430 Ki = 7 nM T08856 C6H5TU 73354941 Ki = 13 nM T08856 CEHB08 73356503 Ki = 364 nM T08856 CUB7V9 76329513 IC50 = 0.4 nM T08856 C5LB0U 78426619 IC50 > 100000 nM T08856 CET6N8 78426757 IC50 > 100000 nM T08856 CKD41G 81689861 IC50 = 2000 nM T08856 COV8I9 86291010 IC50 = 1002 nM T08856 CAB2F5 87349434 Ki = 8700 nM T08856 CVPH63 90663059 Ki = 24000 nM T08856 C6AK3O 90663060 Ki = 17000 nM T08856 CUZD67 90663061 Ki = 9000 nM T08856 CTQ17J 90663062 Ki = 45000 nM T08856 CQGJ90 90663063 Ki = 1000 nM T08856 C0ZH1K 90663064 Ki = 18000 nM T08856 CD53CF 90663065 Ki = 5000 nM T08856 C1A4QT 90663067 Ki = 6000 nM T08856 CLW7Q8 90663069 Ki = 25000 nM T08856 C6JY4Q 90663070 Ki = 40000 nM T08856 C7YU1I 90663071 Ki = 9000 nM T08856 C07RTW 90663072 Ki = 3000 nM T08856 CZ68QM 90663073 Ki = 20000 nM T08856 CVTJ63 90663074 Ki = 5000 nM T08856 C9J8HB 90663075 Ki = 200 nM T08856 C06GRV 90663076 Ki = 100 nM T08856 CF2L9A 90663077 Ki = 48000 nM T08856 CGL0N7 90663078 Ki = 13000 nM T08856 COP05M 90663079 Ki = 12000 nM T08856 C1E5CB 90663080 Ki = 34000 nM T08856 C6IXP4 90663081 Ki = 39000 nM T08856 C0S7NT 90663082 Ki = 10000 nM T08856 C8MOY6 90663083 Ki = 23000 nM T08856 C4NP9W 90663084 Ki = 25000 nM T08856 CD3C8E 90663085 Ki = 18000 nM T08856 C63NOF 90663086 Ki = 20000 nM T08856 CU3LC2 90663087 Ki = 19000 nM T08856 CLCW15 122181996 IC50 > 100000 nM T08856 CT7D4F 122181997 IC50 > 100000 nM T08856 CZO32N 122181998 IC50 > 100000 nM T08856 C40DWG 122181999 IC50 > 100000 nM T08856 CH59PY 127025166 IC50 = 42.2 nM T08856 CM7B5S 127029507 IC50 > 100000 nM T08856 C6HA8I 127029508 IC50 > 100000 nM T08856 CPM3N2 127029509 IC50 = 83.1 nM T08856 C3B9EY 127029510 IC50 > 100000 nM T08856 C89QOM 127043503 IC50 = 228 nM T08856 C9E5YJ 127043505 IC50 = 39 nM T08856 CW1Q3D 127043506 IC50 = 47 nM T08856 C1C7WB 127044036 IC50 = 104.3 nM T08856 CPF6U7 127044139 IC50 = 45.3 nM T08856 CT9B0Q 127044462 IC50 = 59.6 nM T08856 CL3X1A 127044649 IC50 = 226 nM T08856 C8RZ7T 127044651 IC50 = 59 nM T08856 C3I4PT 127044652 IC50 = 81.4 nM T08856 CDX86T 127044818 IC50 = 64.8 nM T08856 C56OJV 127044819 IC50 = 21.3 nM T08856 CYA92R 130282633 IC50 = 2600 nM T08856 CO3QE2 130282636 IC50 = 3700 nM T08856 C4MB7N 132285189 Ki = 7700 nM T08856 CN9D7G 134155756 IC50 > 10000 nM T08856 C7K4PA 135412054 IC50 > 40000 nM T08856 C31VAN 135412231 IC50 > 40000 nM T08856 CHV2U1 135438561 IC50 = 720 nM T08856 CN30DX 135438809 IC50 > 100000 nM T08856 CRAZ20 135485671 IC50 = 3.7 nM T08856 C8R4FB 135546884 IC50 > 40000 nM T08856 C6GR3K 135567051 IC50 = 140 nM T08856 C1MOD4 135567320 IC50 = 600 nM T08856 CYH23I 136054468 IC50 = 22 nM T08856 CZ8DW1 136054472 IC50 = 1000 nM T08856 C9H0DL 136054473 IC50 = 45 nM T08856 CX7MI0 136054475 IC50 = 110 nM T08856 CA5JR6 136054481 IC50 = 14 nM T08856 CO2VU9 136054484 IC50 < 10 nM T08856 CV47JN 136054485 IC50 = 3.9 nM T08856 CZ48WO 136054487 IC50 = 12 nM T08856 CR9CY5 136054490 IC50 = 19 nM T08856 C8FGT0 136054495 IC50 = 56 nM T08856 CGH39U 136054498 IC50 < 10 nM T08856 C2TO7Y 136054508 IC50 = 32 nM T08856 CG70BZ 136054516 IC50 = 1.3 nM T08856 CSM57W 136054520 IC50 = 1.2 nM T08856 CIEW62 136380958 IC50 = 8.9 nM T08856 C9HS7J 137287436 IC50 = 0.82 nM T08856 CQ3GZ0 137632187 Ki = 8500 nM T08856 C4UMY5 137636781 IC50 > 5000 nM T08856 CR8H9Z 137644167 IC50 > 5000 nM T08856 CB8M6U 137646865 IC50 > 5000 nM T08856 CK4LE6 137647628 IC50 = 3500 nM T08856 CXV6J5 137648746 Ki = 19 nM T08856 CZ51XB 137651858 Ki = 3.3 nM T08856 CKH37T 137657100 Ki = 6500 nM T08856 CZB75K 137657128 IC50 > 10000 nM T08856 CC3I9B 137660260 IC50 > 5000 nM T08856 C4H0EM 137661370 IC50 > 5000 nM T08856 C37HMX 137701229 Ki = 2100 nM T08856 C5FWA2 145949488 IC50 = 128 nM T08856 CZS1N7 145949693 IC50 = 113 nM T08856 C6IPV3 145949783 IC50 > 500000 nM T08856 C72LGN 145950074 IC50 = 401100 nM T08856 CU53BP 145950331 IC50 = 270 nM T08856 CY8C4A 145950332 IC50 = 29 nM T08856 CAJ25P 145951291 IC50 > 5000 nM T08856 C3EF7N 145952515 IC50 = 38 nM T08856 CW1GS2 145952760 IC50 > 5000 nM T08856 CFN1R7 145952843 IC50 = 35 nM T08856 CV80WQ 145954107 IC50 = 400 nM T08856 C16VNH 145954604 IC50 = 140 nM T08856 CQF50V 145954863 IC50 = 17 nM T08856 C2HAG8 145955226 IC50 = 483100 nM T08856 CH0ZO5 145955778 IC50 > 5000 nM T08856 CVZ5U7 145955868 IC50 = 117 nM T08856 C8TPR1 145956198 IC50 > 5000 nM T08856 COR96H 145956298 IC50 > 500000 nM T08856 CR8U7Y 145956318 IC50 > 5000 nM T08856 C7R3FE 145956426 IC50 = 198900 nM T08856 CUS0Y9 145957234 IC50 = 1600 nM T08856 C6MHN7 145957508 IC50 > 5000 nM T08856 CQ15DP 145957734 IC50 = 345800 nM T08856 C5K7PV 145958060 IC50 > 5000 nM T08856 CBE02W 145958354 IC50 > 5000 nM T08856 CQL4O0 145959327 IC50 = 832 nM T08856 CG03OE 145959777 IC50 = 172800 nM T08856 CIQ9J2 145960035 IC50 = 298500 nM T08856 CRY63E 145963538 IC50 > 5000 nM T08856 C8UC1T 145963891 IC50 = 90200 nM T08856 CWOF29 145964116 IC50 = 77400 nM T08856 CKD86B 145964366 IC50 = 52500 nM T08856 CI0T9C 145964617 IC50 = 64500 nM T08856 CA94UB 145966060 IC50 = 40400 nM T08856 CL7QD9 145966162 IC50 = 52100 nM T08856 CA80DF 145966420 IC50 = 76500 nM T08856 CNR98O 145966867 IC50 = 39400 nM T08856 CI9JB5 145967177 IC50 = 87500 nM T08856 CJ47BV 145969859 IC50 = 55100 nM T08856 C1R9ES 145971386 IC50 = 24300 nM T08856 CFE1A5 145971595 Ki = 8590 nM T08856 CQ78MP 145971807 IC50 > 100000 nM T08856 CX0JY3 145972073 IC50 > 100000 nM T08856 C1FPG2 145972660 IC50 = 110 nM T08856 CPB91X 145972781 IC50 = 6600 nM T08856 CQ4K0X 145972990 IC50 > 100000 nM T08856 CG4E3F 145973485 IC50 = 46700 nM T08856 CJF73O 145973630 IC50 = 83 nM T08856 CTA0S4 145974193 IC50 = 28200 nM T08856 C52HKA 145974836 IC50 = 43000 nM T08856 CKW8B6 145975533 IC50 = 41500 nM T08856 CTD40B 145975699 IC50 > 100000 nM T08856 CMNS71 145975707 IC50 = 17700 nM T08856 CM6QB0 145976230 IC50 > 100000 nM T08856 CU7HO6 145976282 IC50 = 56100 nM T08856 CW6F2Y 145976412 IC50 = 52500 nM T08856 CX7M9L 145976456 IC50 > 5000 nM T08856 CBD28P 145977013 IC50 = 92100 nM T08856 CPD1B0 145977213 IC50 = 1100 nM T08856 C8CV6O 145977231 IC50 > 100000 nM T08856 C3VOQ8 145978127 IC50 = 89300 nM T08856 C2JQ6E 145978441 IC50 = 33400 nM T08856 C8ZVJ6 145978450 IC50 = 84000 nM T08856 C42JOA 145978615 IC50 > 100000 nM T08856 C2C8QR 153033791 IC50 = 100100 nM T08856 CV10AF 155512426 IC50 = 282 nM T08856 CFHU79 155514943 IC50 = 198 nM T08856 CND4L8 155515645 IC50 = 39700 nM T08856 C0OSL9 155516668 IC50 = 62500 nM T08856 C59YHT 155522902 IC50 = 50 nM T08856 C6RBG9 155527660 IC50 = 25600 nM T08856 CC5FA9 155529859 IC50 > 10000 nM T08856 CQUA53 155531128 IC50 = 5000 nM T08856 C7TP3R 155531151 IC50 > 10000 nM T08856 C5WTE3 155534754 IC50 = 36400 nM T08856 C4VCN3 155535749 IC50 = 30500 nM T08856 C2WCU5 155536887 IC50 = 28200 nM T08856 CO90SD 155541304 IC50 = 65200 nM T08856 CV0ZI3 155542003 IC50 = 48800 nM T08856 CJN8X5 155542058 Ki = 0.6 nM T08856 CH9E0W 155543836 IC50 = 75600 nM T08856 CBSJ86 155544856 IC50 = 48900 nM T08856 CWEG57 155545190 IC50 = 15 nM T08856 CLWS20 155545852 IC50 > 100000 nM T08856 C1FP0M 155548067 IC50 = 172 nM T08856 CM7C1P 155555245 IC50 = 60100 nM T08856 CS62RN 155556052 IC50 = 48100 nM T08856 CJHM29 155557941 IC50 = 35800 nM T08856 CD3M6P 155558654 IC50 = 36800 nM T08856 CPDF57 155558916 IC50 > 100000 nM T08856 C3BA9L 155561798 IC50 = 21 nM T08856 CQ4WE0 155563852 IC50 = 86500 nM T08856 C5U9LI 155569346 IC50 = 2000 nM T08856 CLT4Y6 10138589 Ki = 170 nM T08856 C5U3AO 57394286 IC50 = 138 nM T08856 D00KSS 18411961 IC50 = 1100 nM T08856 D01UNE 44580457 Ki = 38.9 nM T08856 D02ECA 448942 IC50 = 1700 nM T08856 D03SNK 644601 IC50 = 1024 nM T08856 D04VPH 45376872 IC50 > 22000 nM T08856 D05THD 44478925 IC50 = 1000 nM T08856 D07GEL 10344307 Ki = 0.5 nM T08856 D07MJD 44479701 IC50 = 290 nM T08856 D09USO 5277466 IC50 = 52000 nM T08856 D09ZOA 25049753 IC50 = 7 nM T08856 D0A0FY 44479457 IC50 = 72000 nM T08856 D0A4TC 446504 IC50 = 2 nM T08856 D0B3UN 44580458 Ki = 271 nM T08856 D0D7UA 10267279 IC50 = 4 nM T08856 D0H6CK 10160968 Ki = 217 nM T08856 D0K3RC 44294677 IC50 = 8 nM T08856 D0L6ND 10089677 IC50 = 0.39 ug.mL-1 T08856 D0N0FX 19366816 IC50 = 585 nM T08856 D0Q4TA 10044321 IC50 = 260 nM T08856 D0R2BO 194777 IC50 = 0.046 nM T08856 D0S9OL 10155934 IC50 = 620 nM T08856 D0T1FR 44457233 IC50 > 100000 nM T08856 D0V9GS 651854 IC50 = 670 nM T08856 D0W2UK 6914621 Ki = 257 nM T08856 D0XK7G 10445302 Ki = 59 nM T08856 D0Y5IQ 44255320 IC50 = 5000 nM T08856 D0YA8C 10592233 Ki = 560 nM T08856 D0Z2JN 10709191 Ki = 3090.3 nM T92439 D01LCC 17754438 IC50 > 10000 nM T92439 D0A9IY 135564558 IC50 = 1394 nM T92439 D00YPW 135399235 IC50 = 13000 nM T92439 C1B4XD 11992634 IC50 > 2000 nM T92439 CPX16N 11993169 IC50 > 2000 nM T92439 C20VHK 24871823 IC50 = 1400 nM T92439 C6EQG2 24963293 IC50 > 2000 nM T92439 CQU19I 44180409 IC50 = 56 nM T92439 CD52CA 57391118 IC50 > 2000 nM T92439 CWX3N7 59320301 IC50 = 1480 nM T92439 C0EP5I 59341847 IC50 > 10000 nM T92439 CHQ28A 59341978 IC50 > 10000 nM T92439 CBM61I 73293715 IC50 = 963 nM T92439 C9JE6M 75815419 IC50 = 38 nM T92439 C7F6JY 92135987 IC50 > 10000 nM T92439 CQ9X2T 118525749 IC50 > 10000 nM T92439 CA9Z4N 118525753 IC50 > 10000 nM T92439 COM19L 118525755 IC50 > 10000 nM T92439 CCB0S9 118525772 IC50 > 10000 nM T92439 C0SV3H 118525773 IC50 > 10000 nM T92439 CG4Z8E 118525774 IC50 > 10000 nM T92439 CYE6W5 118525795 IC50 > 10000 nM T92439 C8OH0Y 118525801 IC50 > 10000 nM T92439 CP75JF 118525805 IC50 > 10000 nM T92439 CR65SL 118525810 IC50 > 10000 nM T92439 C94ZTQ 118525830 IC50 > 10000 nM T92439 CM8IQ7 118525835 IC50 > 10000 nM T92439 CQ0LU1 118525854 IC50 > 10000 nM T92439 C2PWK5 118534656 IC50 > 10000 nM T92439 C4H2LG 118534683 IC50 > 10000 nM T92439 CRJE23 122185011 IC50 = 7 nM T92439 C62CSI 129051756 IC50 > 10000 nM T92439 C5RFV2 129051760 IC50 > 10000 nM T92439 CH20AQ 129051764 IC50 > 10000 nM T92439 CDJ2V1 129051781 IC50 > 10000 nM T92439 C7AD3Z 129051788 IC50 > 10000 nM T92439 CZ09EG 135418212 IC50 = 4 nM T92439 C7GC0D 135436665 IC50 > 10000 nM T92439 C3R8SE 135457869 IC50 = 1130 nM T92439 CWQG94 135484473 IC50 = 520 nM T92439 CW51OH 135566500 IC50 = 0.4 nM T92439 CR8JM9 135566501 IC50 = 2137.96 nM T92439 CN87GS 135566743 IC50 = 116 nM T92439 CYVU41 135566744 IC50 = 900 nM T92439 CX7I5Z 135721222 IC50 = 1340 nM T92439 CL34KC 135860085 IC50 = 1479.11 nM T92439 CU1W4H 135860086 IC50 = 562.34 nM T92439 C9FO2W 135860090 IC50 = 1318.26 nM T92439 CH5N1M 135860091 IC50 = 269.15 nM T92439 C13QRM 135860092 IC50 = 190 nM T92439 CHT23I 135860093 IC50 = 400 nM T92439 C38XKR 135860094 IC50 = 110 nM T92439 C26ECA 135860095 IC50 = 220 nM T92439 CLM59K 135860101 IC50 = 73 nM T92439 C7QAS6 135873861 IC50 > 1000 nM T92439 CS9DT5 135875901 IC50 = 970 nM T92439 CPM68I 135875902 IC50 = 194.98 nM T92439 C87UJS 135875904 IC50 = 208.93 nM T92439 CVZ12B 135886459 IC50 > 1000 nM T92439 CCH2Z5 135886460 IC50 = 1872 nM T92439 CVP62I 135886467 IC50 = 979 nM T92439 CA53FG 135886468 IC50 = 1603 nM T92439 C6T1EH 135886483 IC50 = 693 nM T92439 C0HJ2E 135886489 IC50 = 165 nM T92439 C09WPF 135886491 IC50 = 431 nM T92439 C3E7IT 135886495 IC50 = 889 nM T92439 C8Q7TD 135886496 IC50 = 466 nM T92439 CTX54Z 135896326 IC50 = 4400 nM T92439 CRP84K 135908600 IC50 = 14 nM T92439 CH6QL0 136059722 IC50 = 970 nM T92439 C2J7ZU 136059723 IC50 = 2050 nM T92439 CN06GO 136059724 IC50 = 3100 nM T92439 C8EA6G 136059725 IC50 = 4200 nM T92439 C31KAG 136059726 IC50 = 7600 nM T92439 C12UMG 136059728 IC50 > 10000 nM T92439 CAH15U 136128521 IC50 = 1858 nM T92439 CW2AZ7 136128560 IC50 = 3421 nM T92439 CBQ31P 136236301 IC50 = 5601 nM T92439 C27HTA 136236310 IC50 = 526 nM T92439 C15POR 136242452 IC50 > 1000 nM T92439 C2C7YL 136242453 IC50 = 297 nM T92439 CLE62X 137179301 IC50 > 10000 nM T92439 C6KYD7 137700754 IC50 > 10000 nM T92439 CM3UF7 137700779 IC50 > 20000 nM T92439 C70YLA 145953136 IC50 > 10000 nM T92439 C0C6FG 145954733 IC50 > 10000 nM T92439 CH7VB3 145957961 IC50 > 10000 nM T92439 C4W2YJ 145961173 IC50 = 579 nM T92439 D06NIT 135564899 IC50 = 50 nM T17221 D06TNL 3278 IC50 = 5000 nM T17221 CZA12R 5141 Ki = 840 nM T17221 C1N8QB 11743150 Ki = 43000 nM T17221 CHX0E8 20731911 Ki = 24300 nM T17221 CF17BR 44300879 Ki = 43000 nM T17221 CEWB31 44300893 Ki = 5800 nM T17221 COJ56C 44300905 Ki = 14700 nM T17221 C3TXO9 44300921 Ki = 360000 nM T17221 C2PJ1R 44413511 IC50 = 13850 nM T17221 COH04A 44413512 IC50 = 32.7 nM T17221 C5UL0A 44413513 IC50 = 24 nM T17221 CIB79M 44413514 IC50 = 13.7 nM T17221 CYR90A 44413516 IC50 = 14.3 nM T17221 C1YL6S 44413517 IC50 = 39.3 nM T17221 CY14GT 44413518 IC50 = 52.1 nM T17221 C7L1EF 44413967 IC50 = 98.9 nM T17221 C4MD6C 60201934 Ki = 135000 nM T17221 C3RWC1 60202091 Ki = 71000 nM T17221 CAX9B5 118706869 Ki = 1470 nM T17221 C7V0QW 118706870 IC50 = 240 nM T17221 C8ABF6 136035723 IC50 = 330 nM T17221 C3JO0P 136035724 IC50 = 180 nM T11192 CK68GT 44580539 IC50 = 4125 nM T11192 D06EHW 11625778 IC50 = 1026 nM T11192 D0W2UK 6914621 Ki = 15 nM T74456 D00JAU 3749 Ki = 0.8 nM T74456 D00NVX 132706 IC50 = 6.9 nM T74456 D04JEE 4946 EC50 > 5011.87 nM T74456 D06UDG 60846 IC50 = 2.7 nM T74456 D0D5SQ 2541 IC50 = 0.69 nM T74456 D0G6SE 172198 Ki = 0.16 nM T74456 D0K0AT 6324663 Ki = 0.17 nM T74456 D0M7TO 60919 IC50 = 32 nM T74456 D0N6RF 65999 IC50 = 0.49 nM T74456 D0T7US 5281037 IC50 = 7.3 nM T74456 D02BBC 6918269 IC50 = 6 nM T74456 D0LI1C 44469321 IC50 > 30000 nM T74456 D0O0JP 9937291 IC50 = 39 nM T74456 D0X2XF 177336 Ki > 10000 nM T74456 D0YS1U 10257882 Ki = 0.8 nM T74456 D00UBK 9851889 IC50 = 1.7 nM T74456 D04AOA 9954408 IC50 = 12 nM T74456 D05UQD 656629 Ki > 10000 nM T74456 D06TZT 132840 Ki = 24 nM T74456 D07LEW 131590 Ki = 29 nM T74456 D0A8HL 3081289 IC50 = 6 nM T74456 D0A9BX 133031 IC50 = 0.2 nM T74456 D0B3CY 121879 IC50 = 3600 nM T74456 D0B5PU 9843631 Ki > 0.0001 nM T74456 D0E3XG 72168 Ki = 1.995 nM T74456 D0F5VB 5311345 Ki = 12 nM T74456 D0GS7N 183134 IC50 = 2.7 nM T74456 D0J2NB 23703120 IC50 = 0.4 nM T74456 D0N5CT 132404 Ki = 20 nM T74456 D0RG2P 9931685 IC50 = 5.6 nM T74456 CN8XG9 156690 Ki > 10 nM T74456 C2J1RE 351037 IC50 > 79000 nM T74456 C1ICH6 1315061 IC50 = 2089.3 nM T74456 C6IPC5 2121575 IC50 = 2570.4 nM T74456 CA61KC 2121583 IC50 = 199 nM T74456 CYIE52 4803452 IC50 = 2187.76 nM T74456 C20VPT 5249743 Ki = 25 nM T74456 CS1W5V 5284633 IC50 = 300 nM T74456 C08QYK 5311348 IC50 > 100000 nM T74456 CX9FV4 7217852 IC50 > 79000 nM T74456 CR1QE5 7217853 IC50 > 79000 nM T74456 C12BHY 7217856 IC50 > 79000 nM T74456 C86MDE 7217859 IC50 > 79000 nM T74456 C9UBG6 7217861 IC50 > 79000 nM T74456 C3XLA7 7217862 IC50 > 79000 nM T74456 C4Y6JF 7217867 IC50 > 79000 nM T74456 CB8NT2 7217870 IC50 > 79000 nM T74456 CT6F3C 7217876 IC50 > 79000 nM T74456 C8PK9D 7217878 IC50 > 79000 nM T74456 CYX8F6 7217879 IC50 > 79000 nM T74456 CH3I6U 7217884 IC50 > 79000 nM T74456 CI92NG 7217887 IC50 > 79000 nM T74456 C17GSL 7217891 IC50 > 79000 nM T74456 C1W3XE 7217912 IC50 > 79000 nM T74456 C8RWT6 7217913 IC50 > 79000 nM T74456 CFOJ16 7217916 IC50 > 79000 nM T74456 C5LZ0X 7217919 IC50 > 79000 nM T74456 CNG45O 7217921 IC50 > 79000 nM T74456 C2PQ8W 7217922 IC50 > 79000 nM T74456 CA7EW6 7217938 IC50 > 79000 nM T74456 CK9X8S 7217939 IC50 > 79000 nM T74456 CT89GV 7217942 IC50 > 79000 nM T74456 C07ZXA 7217944 IC50 > 79000 nM T74456 CUA9S4 7217946 IC50 > 79000 nM T74456 C7AMT6 7217947 IC50 > 79000 nM T74456 CCE5T6 7217950 IC50 > 79000 nM T74456 CW2AT7 7218011 IC50 > 79000 nM T74456 CZI91W 9807029 IC50 = 0.3 nM T74456 C35FCP 9810305 IC50 = 1.8 nM T74456 CT13BE 9823146 IC50 = 16 nM T74456 C91GBS 9824568 IC50 = 11 nM T74456 CPT7L5 9826191 Ki = 0.5012 nM T74456 C8TD2L 9826888 Ki = 0.48 nM T74456 C1I6GK 9850811 IC50 = 1 nM T74456 CIWU91 9850834 IC50 = 1.5 nM T74456 CV07NF 9851082 IC50 = 1 nM T74456 C2C4OM 9852384 IC50 = 1.4 nM T74456 CRP84D 9853391 IC50 = 0.2 nM T74456 C0BH3O 9869504 IC50 = 1.2 nM T74456 C19NOU 9870652 IC50 = 4.5 nM T74456 CG7I2Q 9871837 IC50 = 2 nM T74456 CQ4LC2 9872676 Ki = 3710 nM T74456 C6SHG0 9874508 IC50 = 8.1 nM T74456 CEO03B 9889557 IC50 = 17 nM T74456 CV8A6J 9895212 IC50 = 0.05 nM T74456 CD04YO 9895957 IC50 = 6 nM T74456 C2M4BW 9895984 IC50 = 4 nM T74456 CB0A3I 9896251 IC50 = 13 nM T74456 CI4A8R 9915892 IC50 = 4.2 nM T74456 CY9N3R 9918412 IC50 = 0.2 nM T74456 CP45TL 9939191 Ki = 1.7 nM T74456 C65CYH 9940350 IC50 = 0.5 nM T74456 CJF49M 9960721 IC50 = 1.9 nM T74456 CRL65O 9979771 IC50 = 2.4 nM T74456 C78POU 9981102 IC50 = 7.1 nM T74456 C86VWU 9983135 IC50 = 11.1 nM T74456 C9DAJ6 9984181 IC50 = 0.9 nM T74456 C6HQP8 9984303 IC50 = 2.7 nM T74456 CG0ET4 9987414 IC50 = 0.74 nM T74456 CG8CL2 10004489 Ki = 0.66 nM T74456 CPR16C 10004498 Ki = 0.49 nM T74456 CFTL14 10004646 IC50 = 2.3 nM T74456 C0GTJ4 10005741 Ki = 2.1 nM T74456 CYF76W 10005890 IC50 = 3 nM T74456 C7DIK2 10006693 IC50 = 9.9 nM T74456 CO3PR5 10007306 IC50 = 4.8 nM T74456 CK62VT 10007312 IC50 = 3.3 nM T74456 CA47HV 10007362 IC50 = 0.5 nM T74456 C1J7MU 10007528 IC50 = 18.5 nM T74456 C59NJL 10009984 IC50 = 0.45 nM T74456 CE5H3C 10010071 IC50 = 0.38 nM T74456 CEI76X 10010164 IC50 = 17 nM T74456 C62DQJ 10026681 IC50 = 4.2 nM T74456 C0C5FR 10027175 IC50 = 3.4 nM T74456 CR60PM 10028164 Ki = 4.3 nM T74456 CMX71V 10029695 IC50 = 11.1 nM T74456 CY8KS9 10030086 IC50 = 1.7 nM T74456 CS0BA9 10030110 IC50 = 0.6 nM T74456 C7QU3W 10030426 IC50 = 14.6 nM T74456 CCS31D 10032820 IC50 = 0.32 nM T74456 CE9XN3 10032851 IC50 = 0.5 nM T74456 CY62AG 10032877 IC50 = 0.88 nM T74456 CT6M8J 10032988 IC50 = 0.41 nM T74456 CJ3D0B 10033136 IC50 = 1.9 nM T74456 CY1ZL5 10047444 IC50 = 4530 nM T74456 CDH6Y0 10048770 IC50 = 6.6 nM T74456 CHDB84 10049809 IC50 = 4 nM T74456 C0UX2N 10050044 Ki = 1.3 nM T74456 CS2QT0 10052319 IC50 = 54.5 nM T74456 CUP97S 10052399 IC50 = 0.6 nM T74456 CRJ4P0 10053110 IC50 = 3 nM T74456 C3O6GI 10053367 IC50 = 11.1 nM T74456 CQUS95 10053595 IC50 = 5 nM T74456 CC5GW1 10075811 IC50 = 3.4 nM T74456 CJ9T2Q 10076109 IC50 = 260 nM T74456 CXOA48 10076191 IC50 = 6.4 nM T74456 C6FP7N 10077513 IC50 = 21.9 nM T74456 CRS30P 10078475 IC50 = 28 nM T74456 CCM3D8 10078554 IC50 = 4.3 nM T74456 C3KX6E 10078780 IC50 = 0.94 nM T74456 C6YFD0 10078800 IC50 = 16 nM T74456 CNQ97X 10079601 Ki = 0.65 nM T74456 CTZ5D8 10095241 Ki = 4.3 nM T74456 CC2IQ7 10095683 Ki = 14 nM T74456 CLW5B0 10095986 IC50 = 2.6 nM T74456 CS3W7A 10096683 Ki = 3.9 nM T74456 C8DE6W 10098291 IC50 = 35.7 nM T74456 CS73XM 10100951 IC50 = 0.28 nM T74456 CM9N8U 10101351 IC50 = 0.34 nM T74456 CS7A5F 10101606 IC50 = 0.72 nM T74456 C3F0TU 10101608 IC50 = 0.55 nM T74456 CFN78G 10101690 IC50 = 1.4 nM T74456 CAJ86X 10166561 IC50 = 30 nM T74456 CS7K0L 10209324 IC50 = 2 nM T74456 CKX80Y 10254585 IC50 = 1.3 nM T74456 CW17PJ 10254899 Ki = 8.7 nM T74456 C6HV1R 10255888 IC50 = 446 nM T74456 CG1T0D 10256564 IC50 = 8.5 nM T74456 CUK72W 10256602 IC50 = 0.6 nM T74456 CB93EA 10257293 IC50 = 117 nM T74456 C8KAP3 10257584 IC50 = 5.3 nM T74456 C4ZSK2 10259265 IC50 = 14 nM T74456 CU58CL 10259447 IC50 = 0.36 nM T74456 CEYO10 10259468 IC50 = 0.43 nM T74456 CUA9G7 10259525 IC50 = 1.6 nM T74456 CI0WR6 10259841 IC50 = 1.6 nM T74456 C5LC9E 10280531 IC50 = 24 nM T74456 CO9IC8 10322229 Ki = 1 nM T74456 C1QSM9 10323969 IC50 = 16.6 nM T74456 C6V7WG 10324179 IC50 = 15.9 nM T74456 CH21JQ 10324361 IC50 = 10.1 nM T74456 CMX95I 10324657 IC50 = 12.4 nM T74456 CGV5U6 10324870 IC50 = 8 nM T74456 CHJ4G0 10325267 IC50 = 1.2 nM T74456 CHTL80 10325295 IC50 = 47.9 nM T74456 C9P6UA 10325483 IC50 = 4.9 nM T74456 CZ6ML9 10325767 IC50 = 16.9 nM T74456 CJ9H8M 10327309 IC50 < 0.3 nM T74456 CNZ05L 10327728 IC50 = 24 nM T74456 CW7K4Z 10342301 IC50 = 2.8 nM T74456 C4XZO9 10343090 IC50 = 3.5 nM T74456 CAUB84 10344188 Ki = 0.65 nM T74456 CNOX21 10345537 Ki = 2.7 nM T74456 CLIH83 10349897 IC50 = 4.6 nM T74456 CX1A2T 10350123 IC50 = 4.7 nM T74456 C29KUZ 10366402 Ki = 1.1 nM T74456 CWZ9N7 10367792 IC50 = 7.1 nM T74456 C2NBG6 10369479 IC50 = 40.2 nM T74456 CVD5W6 10369701 IC50 = 5.8 nM T74456 CSUH47 10369867 IC50 = 1.5 nM T74456 CTR4A7 10369902 IC50 = 9 nM T74456 CRVA34 10371118 IC50 = 14.3 nM T74456 C6C8UJ 10371295 IC50 = 159 nM T74456 CK24ZW 10372451 IC50 = 0.44 nM T74456 C8PUW5 10372550 IC50 = 2.2 nM T74456 CAU4G3 10372659 IC50 = 0.76 nM T74456 CWAP07 10372810 IC50 = 5.9 nM T74456 CDJ5M3 10373120 IC50 = 0.96 nM T74456 CNW30P 10390188 Ki = 0.29 nM T74456 C8EBV1 10391038 IC50 = 8.5 nM T74456 C6G3FE 10391950 IC50 = 41.7 nM T74456 C5E8WI 10392378 IC50 = 1.2 nM T74456 C70JVE 10393016 Ki = 10 nM T74456 C9VR4Z 10393086 IC50 = 17.6 nM T74456 C5KEW8 10394727 IC50 = 6 nM T74456 CA07JQ 10394859 IC50 = 6.1 nM T74456 C2WXC5 10395076 IC50 = 0.14 nM T74456 CQB57G 10395335 IC50 = 0.43 nM T74456 C7KY3L 10408794 IC50 = 3.467 nM T74456 C9MRQ6 10414273 IC50 = 8.3 nM T74456 C1XST2 10414338 IC50 = 0.7 nM T74456 C42BDV 10414470 IC50 = 1.4 nM T74456 C5KSE6 10415119 IC50 = 14.5 nM T74456 CB0ZK1 10417195 IC50 = 15 nM T74456 C8QY7E 10417321 IC50 = 3.4 nM T74456 C6FSG7 10439715 IC50 = 0.64 nM T74456 C41IQS 10439819 IC50 = 0.4 nM T74456 CO1V5L 10439837 IC50 = 1 nM T74456 C9GM1L 10439858 IC50 = 8.8 nM T74456 CG1Q7I 10440144 IC50 = 2 nM T74456 C37VCL 10459724 IC50 = 245 nM T74456 C1IL2S 10459992 IC50 = 31 nM T74456 CQ08FG 10460186 IC50 = 23.9 nM T74456 CT61DH 10462573 IC50 = 2.2 nM T74456 C8PCF5 10462598 IC50 = 0.32 nM T74456 CV93HT 10462683 IC50 = 1 nM T74456 CCG2B9 10462933 IC50 = 1.1 nM T74456 CUW9F1 10475382 IC50 = 30 nM T74456 C5IFH8 10478294 IC50 = 4.9 nM T74456 CJ03BC 10478476 IC50 = 44 nM T74456 C7JVR6 10479983 Ki = 0.45 nM T74456 CO83VF 10480064 Ki = 9.6 nM T74456 CT5PQ2 10480309 IC50 = 0.5 nM T74456 CB2QK9 10481196 Ki = 2.7 nM T74456 C1HTM9 10481968 IC50 = 1.4 nM T74456 C8TC5F 10482340 IC50 = 47.8 nM T74456 CL8T2A 10482886 IC50 = 9.8 nM T74456 CQE84K 10483597 IC50 = 4.2 nM T74456 C3XK5L 10504330 Ki = 158 nM T74456 CC8X7L 10507383 Ki = 32 nM T74456 CU1Z3D 10623969 Ki > 10000 nM T74456 CXK68V 10643268 Ki > 10000 nM T74456 CQ42UA 10673314 Ki > 10000 nM T74456 C0GO1E 10674630 Ki = 25 nM T74456 C0IDF4 10695091 Ki > 10000 nM T74456 C1G8FB 10695405 Ki = 398 nM T74456 CZRC03 10697700 Ki = 13 nM T74456 CS2U9K 10697829 Ki = 40 nM T74456 CW90RU 10742620 Ki = 29 nM T74456 C3BYA7 10744859 Ki = 42 nM T74456 CJ7A6K 10763626 IC50 = 9.1 nM T74456 CR2WI1 10764613 Ki = 3162 nM T74456 C5DM4Y 10765881 Ki = 3301 nM T74456 CHP75M 10790260 Ki = 1995 nM T74456 CK4W1Q 10790818 Ki = 381 nM T74456 C5B2HR 10790819 Ki = 402 nM T74456 C9A2FH 10811054 Ki > 10000 nM T74456 C35BIO 10884983 Ki = 80 nM T74456 CV2E4Z 11476710 IC50 = 5.5 nM T74456 CT4KU3 11502835 IC50 = 3 nM T74456 CN4GI8 11561462 IC50 = 60 nM T74456 CVH5U6 11754146 Ki = 0.7 nM T74456 CN5AZ0 11754586 Ki = 12 nM T74456 CN9W0D 11757112 IC50 = 34.6 nM T74456 CJ6D4Q 11757216 IC50 = 198 nM T74456 C0G7ME 11757908 IC50 = 104 nM T74456 CL0X3B 11758329 IC50 = 70 nM T74456 CSQ3P5 11758341 IC50 = 8 nM T74456 CUJ7E0 11758470 IC50 = 17.8 nM T74456 CDGF69 11765177 IC50 = 3.3 nM T74456 CD7E5Q 11765454 IC50 = 1.5 nM T74456 C9I0HX 11765560 IC50 = 0.84 nM T74456 CZ2C1H 11801362 Ki = 32 nM T74456 C9ZEC8 12005825 IC50 > 79000 nM T74456 C1D7HW 12005898 IC50 > 79000 nM T74456 C4K8HT 12005992 IC50 > 79000 nM T74456 CD45PU 14952903 IC50 = 440 nM T74456 CQZ71Y 15222070 IC50 = 2 nM T74456 CG5XH2 15222092 IC50 = 2 nM T74456 CBPL06 15222094 IC50 = 2 nM T74456 CO5V6R 15222101 IC50 = 10 nM T74456 CO71QD 15222103 IC50 = 6 nM T74456 CF57HL 15292111 IC50 = 10 nM T74456 CX75ZV 15292112 IC50 = 12 nM T74456 CG29NO 15292113 IC50 = 0.71 nM T74456 CSK27N 15818746 IC50 = 9 nM T74456 CV40ST 15818748 IC50 = 1 nM T74456 CB78RO 16130452 Ki > 100000 nM T74456 C0A9WY 16194671 IC50 > 79000 nM T74456 C6J4NC 16805942 IC50 > 79000 nM T74456 C21UXH 16832372 IC50 > 79000 nM T74456 C8NGJ0 18004820 IC50 = 21 nM T74456 C9IP8D 18572334 IC50 > 79000 nM T74456 CK2L9R 18572335 IC50 > 79000 nM T74456 CO48HV 18572337 IC50 = 60100 nM T74456 CC70BA 18572338 IC50 > 79000 nM T74456 CMG17E 18572343 IC50 > 79000 nM T74456 CQ3ZV0 18572352 IC50 > 79000 nM T74456 CZ2FW0 18572378 IC50 > 79000 nM T74456 COP52X 18572379 IC50 > 79000 nM T74456 CAJH61 18572382 IC50 > 79000 nM T74456 CNKA87 18572395 IC50 > 79000 nM T74456 CL94NS 18654313 IC50 = 661 nM T74456 CA82PW 19008901 IC50 = 96 nM T74456 CT7ED5 19008935 IC50 = 238 nM T74456 CAG89Z 19102815 IC50 = 150 nM T74456 C8BLT0 19430442 IC50 = 0.28 nM T74456 CVL4G0 19430458 IC50 = 0.74 nM T74456 C60YHR 19430462 IC50 = 0.35 nM T74456 CRC30I 19430475 IC50 = 0.57 nM T74456 CVF5K9 19430479 IC50 = 0.6 nM T74456 CSD1U8 19919870 IC50 = 884 nM T74456 C2KQ7M 19939495 IC50 = 110 nM T74456 CBZ9S7 20081627 IC50 = 1.8 nM T74456 C5FZX8 20747575 IC50 = 8 nM T74456 C0X4NY 21840324 IC50 = 30 nM T74456 CK4H2W 21840429 IC50 = 600 nM T74456 C8JZT4 22574723 IC50 = 1.3 nM T74456 CFP01R 24828743 Ki = 549.54 nM T74456 C0TR3U 25190005 Ki = 5.012 nM T74456 C8TX1U 42281625 IC50 > 79000 nM T74456 CE69MC 44210864 IC50 = 3 nM T74456 C5FDC2 44254496 Ki = 141.25 nM T74456 CR28CF 44264673 IC50 = 22 nM T74456 C5J6NY 44277442 IC50 = 6.9 nM T74456 C4VK6Q 44277443 IC50 = 5.7 nM T74456 CNX92H 44277461 IC50 = 21.4 nM T74456 CE8TQ6 44277549 IC50 = 10.6 nM T74456 CYIF37 44277567 IC50 = 4.4 nM T74456 CM1K2L 44277573 IC50 = 0.9 nM T74456 CK81TH 44277574 IC50 = 5.09 nM T74456 C97IVT 44277593 IC50 = 9.6 nM T74456 CSC65I 44277594 IC50 = 6 nM T74456 C9TP0H 44277677 IC50 = 4 nM T74456 C93WRI 44277871 IC50 = 4.9 nM T74456 C7VM0B 44285157 IC50 = 100 nM T74456 CO2J0U 44285177 IC50 = 20 nM T74456 CH10OD 44285178 IC50 = 3 nM T74456 CGA4L5 44285212 IC50 = 1400 nM T74456 CV3WH8 44285267 IC50 = 0.9 nM T74456 CCF0T1 44285327 IC50 = 8 nM T74456 C8MR7S 44285370 IC50 = 4 nM T74456 CQD25K 44285371 IC50 = 300 nM T74456 C7VY6C 44285372 IC50 = 2 nM T74456 CJSW19 44301981 IC50 = 44 nM T74456 C4MH6O 44311071 IC50 = 1 nM T74456 C04OWQ 44311072 IC50 = 0.1 nM T74456 CVXU13 44311073 IC50 = 0.1 nM T74456 C64VDR 44311074 IC50 = 0.2 nM T74456 C3O6SW 44311182 IC50 = 0.5 nM T74456 CCD7K5 44311183 IC50 = 0.8 nM T74456 CDC7V8 44311184 IC50 = 0.6 nM T74456 CYSE79 44311185 IC50 = 0.3 nM T74456 CFO20B 44311289 IC50 = 0.2 nM T74456 C5FI1X 44311342 IC50 = 10 nM T74456 CHW83V 44311406 IC50 = 20 nM T74456 C37PFG 44311412 IC50 = 0.2 nM T74456 CAK8C2 44311413 IC50 = 0.2 nM T74456 CHJP87 44311414 IC50 = 0.1 nM T74456 C3WZY9 44311415 IC50 = 0.1 nM T74456 COTX54 44311428 IC50 = 10 nM T74456 C8C5HR 44311429 IC50 = 40 nM T74456 CW7V8A 44311434 IC50 = 0.1 nM T74456 CT6A4H 44311435 IC50 = 0.1 nM T74456 C7FH8G 44311436 IC50 = 3 nM T74456 C5P6NM 44311449 IC50 = 10 nM T74456 CWVO75 44311450 IC50 = 10 nM T74456 CL68EO 44311451 IC50 = 2 nM T74456 C3H1MD 44311452 IC50 = 0.5 nM T74456 C3F6SU 44311453 IC50 = 0.4 nM T74456 C6Q0UC 44311454 IC50 = 0.3 nM T74456 C7SD4Z 44311455 IC50 = 0.1 nM T74456 CKT0U8 44311456 IC50 = 0.2 nM T74456 C5HPL4 44311472 IC50 = 100 nM T74456 C23KJT 44311496 IC50 = 8 nM T74456 C9CY1G 44311497 IC50 = 2 nM T74456 CC9Y6E 44311498 IC50 = 3 nM T74456 CL9Z1B 44311499 IC50 = 2 nM T74456 CRF13T 44311537 IC50 = 0.3 nM T74456 CKI10X 44311538 IC50 = 0.8 nM T74456 COI20G 44311543 IC50 = 10 nM T74456 C4FAK2 44311557 IC50 = 0.3 nM T74456 CB41MY 44311558 IC50 = 0.6 nM T74456 C3X1AL 44311567 IC50 = 9 nM T74456 CY7DG6 44311568 IC50 = 20 nM T74456 C1XC8Q 44311569 IC50 = 20 nM T74456 CD4ZM5 44311571 IC50 = 9 nM T74456 C5UBK7 44311580 IC50 = 0.1 nM T74456 CX90KA 44311581 IC50 = 0.2 nM T74456 CT05AS 44311582 IC50 = 0.2 nM T74456 CUAI35 44311583 IC50 = 2 nM T74456 CTP18U 44311584 IC50 = 8 nM T74456 C04GME 44311607 IC50 = 6 nM T74456 C0R6QJ 44311609 IC50 = 30 nM T74456 C5LJ8A 44311616 IC50 = 9 nM T74456 CSH0R1 44311617 IC50 = 0.6 nM T74456 C92KSW 44311618 IC50 = 0.6 nM T74456 CPGV60 44311619 IC50 = 0.4 nM T74456 CSE80D 44311635 IC50 = 0.9 nM T74456 C6CQ3Y 44311636 IC50 = 20 nM T74456 CLT7J0 44311638 IC50 = 30 nM T74456 CXZ1Y2 44311648 IC50 = 2 nM T74456 CX89YT 44311650 IC50 = 6 nM T74456 CU4HB9 44311662 IC50 = 2 nM T74456 C0I8FS 44311663 IC50 = 2 nM T74456 CT1X8Z 44311664 IC50 = 10 nM T74456 CR7Q4V 44311675 IC50 = 0.3 nM T74456 C3X7ZI 44311676 IC50 = 0.1 nM T74456 C8SY2D 44311681 IC50 = 2 nM T74456 C46NML 44311683 IC50 = 0.4 nM T74456 CP7CY2 44311688 IC50 = 10 nM T74456 CJ9A7D 44311715 IC50 = 0.2 nM T74456 C07CUQ 44311735 IC50 = 0.8 nM T74456 CBW43X 44311736 IC50 = 0.3 nM T74456 CPX02A 44311738 IC50 = 5 nM T74456 CJ2N1I 44311739 IC50 = 3 nM T74456 CA1Y6I 44311752 IC50 = 0.3 nM T74456 CAB87G 44311753 IC50 = 0.2 nM T74456 C8VU6N 44311754 IC50 = 1 nM T74456 C8UXN7 44311755 IC50 = 3 nM T74456 CFZE67 44311758 IC50 = 2 nM T74456 C29QVB 44311775 IC50 = 3 nM T74456 CKF7H2 44311776 IC50 = 3 nM T74456 CT6WL4 44312565 IC50 = 0.47 nM T74456 CQWN95 44312700 IC50 = 44 nM T74456 CLV28B 44314761 IC50 = 0.84 nM T74456 CUIL91 44314780 IC50 = 7.2 nM T74456 CD28FL 44314822 IC50 = 1.2 nM T74456 CJS04N 44314823 IC50 = 0.89 nM T74456 CXDG91 44315057 IC50 = 26.5 nM T74456 C6XVW9 44315058 IC50 = 15 nM T74456 C08CHF 44315059 IC50 = 85 nM T74456 C4VD7T 44315060 IC50 = 33 nM T74456 C2JM6E 44315078 IC50 = 1.9 nM T74456 CF89XK 44315144 IC50 = 1.5 nM T74456 C8S9UP 44315180 IC50 = 12 nM T74456 CH0ZF3 44315282 IC50 = 5.8 nM T74456 C1STV6 44315304 IC50 = 14.7 nM T74456 CTD3M0 44315344 IC50 = 65 nM T74456 CJ4SK0 44315349 IC50 = 18 nM T74456 C8QAE0 44315350 IC50 = 59 nM T74456 CH9Q0J 44315351 IC50 = 1.6 nM T74456 C6BRL3 44316861 IC50 = 298 nM T74456 C9G4AK 44316916 IC50 = 2.9 nM T74456 CWOM31 44317214 IC50 = 48.3 nM T74456 CUY7K1 44325313 Ki = 2.9 nM T74456 C0OYS5 44341922 IC50 = 6 nM T74456 CU14EM 44341923 IC50 = 270 nM T74456 CIQ3Y5 44341924 IC50 = 60 nM T74456 C6AQK3 44341946 IC50 = 24 nM T74456 CK3L7P 44342142 IC50 = 200 nM T74456 C3W0UX 44348523 IC50 = 1 nM T74456 CSO26P 44372686 IC50 = 4 nM T74456 CTRJ86 44372814 IC50 = 15 nM T74456 CQ46VS 44373238 IC50 = 8600 nM T74456 CI8HL6 44404967 IC50 = 13 nM T74456 C4DL5C 44469677 IC50 > 10000 nM T74456 CF31QH 44475015 Ki = 15.85 nM T74456 CB31ST 44726831 IC50 > 79000 nM T74456 C65RAJ 45102601 Ki = 1.259 nM T74456 CG3B8F 45102750 Ki = 0.69 nM T74456 CY05QP 45140560 Ki = 0.7 nM T74456 CG6H2E 45140755 Ki = 31.6 nM T74456 CL2B7W 45140756 Ki = 12.8 nM T74456 CIE1Z6 45141357 Ki = 0.5 nM T74456 CV9GP5 45141358 Ki = 58.2 nM T74456 C0C3AG 45141588 Ki = 3.8 nM T74456 C89QTJ 46184983 IC50 = 12.7 nM T74456 C2R8WH 46232959 IC50 = 288 nM T74456 C3Q6DN 46233002 IC50 > 10000 nM T74456 CH41CI 46835118 IC50 > 79000 nM T74456 C5LJ0V 46835120 IC50 > 79000 nM T74456 CSBO37 46835124 IC50 > 79000 nM T74456 C02ICV 46880542 Ki >= 250 nM T74456 CU2SF8 46880543 Ki >= 250 nM T74456 C6EFX7 46905014 IC50 > 79000 nM T74456 CCUA93 46905018 IC50 > 79000 nM T74456 C85DJM 46905020 IC50 > 79000 nM T74456 CBNT43 46905022 IC50 > 79000 nM T74456 CH20YA 46905025 IC50 > 79000 nM T74456 CWER26 46905028 IC50 > 79000 nM T74456 CD3CK1 46905029 IC50 > 79000 nM T74456 CU6D2Q 46905034 IC50 > 79000 nM T74456 CWY35N 46905037 IC50 > 79000 nM T74456 CP3M2F 46905038 IC50 > 79000 nM T74456 CD47WG 46910493 IC50 = 3.7 nM T74456 C3Y5WG 46910494 IC50 = 22.5 nM T74456 C6ZUA1 46910495 IC50 = 2.6 nM T74456 C4EOT6 46910581 IC50 = 78 nM T74456 CBAG18 46910582 IC50 = 57.6 nM T74456 CF7ID9 46910583 IC50 = 214 nM T74456 C83NXB 46935596 Ki > 10000 nM T74456 CQK7D4 49787115 IC50 > 79000 nM T74456 C86OIB 49787117 IC50 > 79000 nM T74456 CL3D2B 49787119 IC50 > 79000 nM T74456 CP5M7Y 49787120 IC50 > 79000 nM T74456 CW9G1R 49842899 IC50 > 79000 nM T74456 CVC2N3 49842902 IC50 > 79000 nM T74456 C9T3AM 49842903 IC50 > 79000 nM T74456 CQ6V4E 49842905 IC50 > 79000 nM T74456 C62CDL 49842908 IC50 > 79000 nM T74456 C6F2KY 53309128 IC50 = 10.5 nM T74456 C9SA4X 53309129 IC50 = 13.3 nM T74456 C07WMK 53309130 IC50 = 10.2 nM T74456 CLV60X 53309271 IC50 = 8.2 nM T74456 C0SL6H 53309272 IC50 = 202 nM T74456 CBPQ05 53309273 IC50 = 15.7 nM T74456 CR3N6U 53309274 IC50 = 6.8 nM T74456 CA97CK 53309275 IC50 = 16.9 nM T74456 CI6KE2 53309404 IC50 = 3.5 nM T74456 C1EM8J 53309405 IC50 = 748 nM T74456 C0EH4S 53309406 IC50 = 5.2 nM T74456 CG6Z4R 53317942 IC50 = 22 nM T74456 C3U5VH 53319274 Ki = 10 nM T74456 C16BWL 53837978 IC50 = 1100 nM T74456 C0EM7R 54178446 IC50 = 7.6 nM T74456 CG2Z0P 54578725 IC50 = 2.6 nM T74456 CQ3K9X 54693559 IC50 = 0.17 nM T74456 CE75ZL 54768659 IC50 = 2000 nM T74456 CB6FV2 54768660 IC50 = 1600 nM T74456 CBY5V7 54768661 IC50 = 1900 nM T74456 C8ZC6M 54768876 IC50 = 3900 nM T74456 CV4L6Q 54768877 IC50 = 5800 nM T74456 CE8LU3 54771778 IC50 = 2300 nM T74456 C9DMZ4 56964910 Ki > 10000 nM T74456 CW9IF2 57380213 IC50 = 52.5 nM T74456 C20CLX 57380412 IC50 = 2.4 nM T74456 CG09ZX 57380413 IC50 = 326 nM T74456 C19NLI 57380414 IC50 = 4.3 nM T74456 CQ5IJ3 57380415 IC50 = 30.6 nM T74456 C2AVN8 57380416 IC50 = 30.8 nM T74456 CZRA28 57380647 IC50 = 1.3 nM T74456 C5Y1TQ 57380648 IC50 = 106 nM T74456 C52XFK 57380649 IC50 = 198 nM T74456 C1L5WH 60148656 IC50 = 0.7 nM T74456 C5RH7K 60165459 IC50 = 6 nM T74456 CX60UI 67472601 Ki > 10000 nM T74456 C8HRB4 70682146 IC50 = 0.9 nM T74456 CGE5V6 70682147 IC50 = 209 nM T74456 CO58GY 70684248 IC50 = 410 nM T74456 C69ZRA 70684421 IC50 = 630.96 nM T74456 C1PNK9 70686409 IC50 = 19.7 nM T74456 C3GC6L 70686410 IC50 = 1.3 nM T74456 CLH90A 70688502 IC50 = 118.5 nM T74456 CPYZ87 70688503 IC50 = 96.8 nM T74456 C1Q2KU 70688504 IC50 = 37.6 nM T74456 C65DSI 70688681 IC50 = 245 nM T74456 CWP1K8 70690562 IC50 = 78.3 nM T74456 CXK5O2 70690743 IC50 = 117.49 nM T74456 C47THE 70694919 IC50 = 23.99 nM T74456 CCQK74 71456693 IC50 > 79000 nM T74456 CGM32X 71462076 IC50 > 79000 nM T74456 CU73LD 71465043 Ki = 10 nM T74456 CA95RY 71520500 IC50 = 6.8 nM T74456 CGTO05 71520501 IC50 = 7 nM T74456 CQ80JF 71521194 IC50 = 593 nM T74456 CC3F8V 71521195 IC50 = 24.4 nM T74456 CP4W1D 71521196 IC50 = 19.8 nM T74456 CHN49X 71521298 IC50 = 348 nM T74456 C94MCT 71521299 IC50 = 19.4 nM T74456 C9C2NZ 71521300 IC50 = 41 nM T74456 CM79CL 71521301 IC50 = 37.7 nM T74456 CO01SV 71521302 IC50 = 5.1 nM T74456 C5V9UO 71521416 IC50 = 13.5 nM T74456 C89DQL 71521417 IC50 = 94.1 nM T74456 CAT53R 71521418 IC50 = 29.3 nM T74456 CJU56D 71521419 IC50 = 67.4 nM T74456 CM96IV 71521503 IC50 = 36.9 nM T74456 CFA2P7 71521504 IC50 = 81.6 nM T74456 CGN94D 71521505 IC50 = 63.8 nM T74456 CA0K3Z 71521506 IC50 = 45.2 nM T74456 CW1G9U 71521507 IC50 = 250 nM T74456 CPC40O 71521585 IC50 = 63.4 nM T74456 CY4R3B 71623945 IC50 = 293.1 nM T74456 C46YXS 71652853 IC50 = 0.3467 nM T74456 C08SFE 71652855 IC50 = 331.13 nM T74456 CR9B4X 71652857 IC50 = 4.266 nM T74456 CXW1A5 71653008 IC50 = 501.19 nM T74456 CBN4R6 71653151 IC50 = 1698.24 nM T74456 CD79SI 71653304 IC50 = 0.912 nM T74456 C62BDU 71653456 IC50 = 2.884 nM T74456 C8VJ6U 71653747 IC50 = 831.76 nM T74456 CNZ74D 71653749 IC50 = 707.95 nM T74456 CKI9F2 71654379 IC50 = 6456.54 nM T74456 CS0XF8 71654381 IC50 = 42.66 nM T74456 C3HRL4 71717081 IC50 = 416.87 nM T74456 CWH6T3 72548703 IC50 = 0.47 nM T74456 C6EG3T 72697299 Ki > 10000 nM T74456 CIQ29F 72697441 Ki > 10000 nM T74456 CN2GV9 72697443 Ki = 1584.89 nM T74456 CS3I2T 73346386 IC50 = 3 nM T74456 CP2ZR0 73346387 IC50 = 1008 nM T74456 C5L6PQ 73347892 IC50 = 0.4 nM T74456 C4COR6 73347893 IC50 = 0.1 nM T74456 CXYJ62 73349423 IC50 = 1430 nM T74456 CEOK17 73349424 IC50 = 20 nM T74456 CJ6VY2 73350990 IC50 = 115 nM T74456 C2LTU4 73350991 IC50 = 4.9 nM T74456 C7KAB4 73352461 IC50 = 1345 nM T74456 CT1XL6 73352589 Ki > 10000 nM T74456 C9ZC5N 73353933 IC50 = 10 nM T74456 CG71DK 73353934 IC50 = 0.3 nM T74456 CRGQ95 73355474 IC50 = 11 nM T74456 CCEA97 73355475 IC50 = 1.2 nM T74456 CB9DV4 73357016 IC50 = 3.9 nM T74456 CU53JN 73357017 IC50 = 13 nM T74456 C6HJS2 73357018 IC50 = 39 nM T74456 CT9AW2 75031588 Ki = 39.81 nM T74456 C35STH 76310606 IC50 = 128 nM T74456 C18EZQ 76310607 IC50 > 10000 nM T74456 C7DE3L 76310608 IC50 > 10000 nM T74456 CIR72S 76310609 IC50 = 1000 nM T74456 C7IOX1 76310610 IC50 = 60 nM T74456 C2VG1F 76315849 IC50 = 25.4 nM T74456 C9QN4E 76317814 IC50 > 10000 nM T74456 CP7E1N 76317815 IC50 = 97 nM T74456 CS1C9M 76319527 IC50 = 6.1 nM T74456 CD36HB 76321525 IC50 = 23 nM T74456 CZ2I6V 76324571 IC50 = 2.5 nM T74456 CR12QV 76325125 IC50 > 10000 nM T74456 CH1W8N 76325126 IC50 = 1690 nM T74456 C2GY6R 76328690 IC50 = 85 nM T74456 CFNP75 76330043 IC50 = 3.3 nM T74456 C2Q9LU 76330395 IC50 = 9.6 nM T74456 CP4CK9 76333686 IC50 = 29.6 nM T74456 CM4D5H 76333687 IC50 = 2.5 nM T74456 C06XHV 86727577 EC50 = 5100 nM T74456 CK4O2F 87218352 Ki = 50.12 nM T74456 C8O1QX 87218371 Ki = 398.11 nM T74456 C92GXJ 87218373 Ki = 1.259 nM T74456 C8I9AL 87218397 Ki = 630.96 nM T74456 CUT8K1 87218444 Ki = 100 nM T74456 C4BQD9 87218492 Ki = 5.012 nM T74456 C8NEO1 87218514 Ki = 1.259 nM T74456 CR45XW 87218658 Ki = 6.31 nM T74456 C3OGP8 87218678 Ki = 39.81 nM T74456 C0DUB7 87218698 Ki = 5.012 nM T74456 C89OAU 87218826 Ki = 251.19 nM T74456 C1UMO7 87218835 Ki = 31.62 nM T74456 CLIT52 87218933 Ki = 125.89 nM T74456 C2L9SX 87218987 Ki = 19.95 nM T74456 CE09GY 87219028 Ki = 6.31 nM T74456 CREO05 87219032 Ki = 0.7943 nM T74456 C4FML3 87219128 Ki = 125.89 nM T74456 CM96JH 87219174 Ki = 2.512 nM T74456 CM58JI 90219582 EC50 = 5500 nM T74456 C2OQC3 118719137 Ki = 2230 nM T74456 CB0QI8 127026027 IC50 = 87.8 nM T74456 CU0J4F 127026040 IC50 = 69.4 nM T74456 C9QA0N 127026041 IC50 = 67.5 nM T74456 C63KTY 127026042 IC50 = 53.5 nM T74456 C8X0UC 127026043 IC50 = 44 nM T74456 CXN21Q 127026058 IC50 = 347 nM T74456 C4PWU0 127026336 IC50 = 30.7 nM T74456 CFY04E 127026337 IC50 = 93 nM T74456 C5YIM7 127026338 IC50 = 90 nM T74456 C04OWP 127028595 IC50 = 140 nM T74456 CSO5F2 127028617 IC50 = 363 nM T74456 C1OFQ0 127028618 IC50 = 161 nM T74456 C9OW0V 127028619 IC50 = 439 nM T74456 CKY51I 127028620 IC50 = 390 nM T74456 CVKG08 127028930 IC50 = 73.7 nM T74456 CHP7W8 127029201 IC50 = 32.9 nM T74456 CWSI52 127029202 IC50 = 3.9 nM T74456 CH5B3Y 127029203 IC50 = 26.1 nM T74456 CS10YM 127029204 IC50 = 36.9 nM T74456 C36HRE 127030653 EC50 = 1.4 nM T74456 CY0CD4 127030942 Ki = 0.71 nM T74456 C9DO8P 127031265 EC50 = 2.042 nM T74456 CXAG39 127031544 EC50 = 2.344 nM T74456 CHU1J9 127031847 Ki = 9 nM T74456 CEJQ23 127034739 IC50 = 342.8 nM T74456 CU8XB9 127034740 IC50 = 366.3 nM T74456 C5UE4D 127034756 IC50 = 160 nM T74456 CWH4T7 127034757 IC50 = 152 nM T74456 C5E4BU 127034758 IC50 = 13 nM T74456 CGK8W6 127034873 IC50 = 1.1 nM T74456 C7B0JQ 127034874 IC50 = 104 nM T74456 CV4KS1 127034875 IC50 = 93.9 nM T74456 CVK0D7 127034876 IC50 = 106.5 nM T74456 CGVR16 127034901 IC50 = 31 nM T74456 CA15SF 127034903 IC50 = 161.1 nM T74456 CQI70D 127034904 IC50 = 738.4 nM T74456 CF9S8X 127034905 IC50 = 1117.3 nM T74456 CT31NI 127034916 IC50 = 94 nM T74456 CPL08Z 127034917 IC50 = 95 nM T74456 CU39OI 127034918 IC50 = 373 nM T74456 C64HFO 127034919 IC50 = 341 nM T74456 CN7DB6 127034920 IC50 = 57.4 nM T74456 CQOV56 127034921 IC50 = 7.3 nM T74456 CRF7J1 127034922 IC50 = 6.3 nM T74456 CZ61LK 127034966 EC50 > 5011.87 nM T74456 CA0SN5 127034967 EC50 > 5011.87 nM T74456 C5XM0K 127035067 IC50 = 47 nM T74456 C1QJ0V 127035068 IC50 = 201 nM T74456 CBC74Y 127035069 IC50 = 419 nM T74456 C67FNJ 127035070 IC50 = 28 nM T74456 CL01XK 127035082 IC50 = 50 nM T74456 CP6T3J 127035083 IC50 = 81 nM T74456 CJHG08 127035084 IC50 = 56 nM T74456 CLJ94G 127035085 IC50 = 8 nM T74456 CRN65G 127035219 IC50 = 217 nM T74456 C83ZIH 127035246 IC50 = 3.5 nM T74456 CQV63D 127035247 IC50 = 1368.1 nM T74456 C6JTW5 127035248 IC50 = 609.2 nM T74456 C9RCI8 127035249 IC50 = 699.3 nM T74456 C3AJ4Z 127035263 IC50 = 61.2 nM T74456 C7OE8P 127035264 IC50 = 2.7 nM T74456 C6CP8U 127035265 IC50 = 1.4 nM T74456 CE07IC 127035379 IC50 = 42 nM T74456 C6DU4R 127035380 IC50 = 76 nM T74456 C9S4JW 127035381 IC50 = 671.4 nM T74456 C75KYB 127035391 IC50 = 788.4 nM T74456 C2NX4L 127035392 IC50 = 486.8 nM T74456 CP30HO 127035393 IC50 = 621.6 nM T74456 C3XWN4 127035410 IC50 = 16 nM T74456 CHN1I9 127035514 IC50 = 156.8 nM T74456 CIKB36 127035515 IC50 = 38.9 nM T74456 CA9FD3 127035544 IC50 = 37 nM T74456 CF6X3E 127035545 IC50 = 92 nM T74456 CHWP78 127035557 IC50 = 503.3 nM T74456 C2SI6O 127035558 IC50 = 87.2 nM T74456 CRAX67 127035715 IC50 = 40.4 nM T74456 C1BZJ5 127035716 IC50 = 23 nM T74456 CZM6R9 127035717 IC50 = 5 nM T74456 C5ED6S 127035757 IC50 = 7 nM T74456 CD0T4M 127036102 IC50 = 19.5 nM T74456 CW6Z5T 127036103 IC50 = 90.5 nM T74456 C5E6QH 127036104 IC50 = 1534.5 nM T74456 C2E0ZQ 127036105 IC50 = 495.8 nM T74456 C3WQD1 127036106 IC50 = 128.6 nM T74456 CNX0J3 127036107 IC50 = 57.9 nM T74456 CR1YG9 127036108 IC50 = 70 nM T74456 CQLC17 127036294 IC50 = 1536.6 nM T74456 C63ZGR 127036297 IC50 = 214.4 nM T74456 CZN92T 127036865 IC50 = 82 nM T74456 C0KJO7 127036866 IC50 = 73.3 nM T74456 C19VDE 127036867 IC50 = 53.9 nM T74456 C24HFS 127036868 IC50 = 549.8 nM T74456 CPQB01 127037496 IC50 = 465 nM T74456 CEQS03 127037497 IC50 = 385 nM T74456 CW8QT1 137527725 IC50 >= 10 nM T74456 C2ND9V 137532858 IC50 = 1.6 nM T74456 C7KD9N 142533975 IC50 = 2.2 nM T74456 C6Z9HB 142534004 IC50 = 38 nM T74456 C8UL6O 142534045 IC50 = 0.7 nM T74456 C9UR5L 142534050 IC50 = 2 nM T74456 CKV4L6 142534121 IC50 = 2.1 nM T74456 C5ZXV2 142534141 IC50 = 1.2 nM T74456 C9AS2D 142534170 IC50 = 32 nM T74456 CXJ8M1 142534183 IC50 = 4.7 nM T74456 C9HAT3 142534191 IC50 = 5.6 nM T74456 CGM6C1 145925549 EC50 = 44 nM T74456 CF8I6Q 145948674 Ki = 13 nM T74456 CQBU72 145952582 Ki = 317 nM T74456 CI2M1Q 145957579 Ki = 24838 nM T74456 CKGV06 145957897 Ki = 1.35 nM T74456 C8QL0G 145981239 IC50 = 1.8 nM T74456 CQB9O0 145987183 IC50 = 70 nM T74456 CG6KB7 155512629 Ki = 7.943 nM T74456 C9KP4F 155513439 Ki = 79.43 nM T74456 C1HOG5 155514738 Ki = 10 nM T74456 CN7Z5E 155516694 Ki = 199.53 nM T74456 C1PUC8 155517399 IC50 = 2.2 nM T74456 C21TUL 155520317 Ki = 125.89 nM T74456 CX1YU9 155522135 Ki = 398.11 nM T74456 C30EFX 155523092 Ki = 125.89 nM T74456 C7WI9L 155526996 Ki = 31.62 nM T74456 C1G7LY 155529942 Ki = 50.12 nM T74456 CVXJ96 155533580 Ki = 63.1 nM T74456 CNV2A8 155535176 Ki = 158.49 nM T74456 C5D3AP 155542482 IC50 = 1.5 nM T74456 CFM26N 155547799 Ki = 50.12 nM T74456 C5AF2L 155551279 EC50 = 17 nM T74456 C1RUT3 155552503 Ki = 31.62 nM T74456 CUE8Y9 155557693 Ki = 15.85 nM T74456 CS7ZV8 155565351 Ki = 79.43 nM T74456 D00LWG 46880545 Ki = 0.7 nM T74456 D04SVT 9829012 IC50 = 0.1 nM T74456 D05NXX 7217941 IC50 > 79000 nM T74456 D06DRC 45141142 Ki = 0.3 nM T74456 D06PJZ 45140373 Ki = 0.6 nM T74456 D07EWK 46880541 Ki = 0.4 nM T74456 D0A4NO 6603900 IC50 = 1.1 nM T74456 D0D1FT 108185 IC50 = 2 nM T74456 D0K2EX 9804984 Ki = 10000 nM T74456 D0L3PY 123814 Ki = 407.38 nM T74456 D0M5ZE 5311416 Ki < 10000 nM T74456 D0MH1K 9935096 IC50 = 4.9 nM T74456 D0N2WA 46880540 Ki = 0.8 nM T74456 D0O0SH 9932483 IC50 = 6.5 nM T74456 D0O1YO 45140942 Ki = 0.4 nM T74456 D0PB5Q 3132 Ki > 10000 nM T74456 D0U7QE 45140941 Ki = 0.7 nM T74456 D0XO1T 46880544 Ki = 0.6 nM T74456 D0Z7AF 10031067 IC50 = 2.1 nM T38529 D06FEA 5280360 Ki = 1.03 nM T38529 D0WL5V 9867642 Ki = 136 nM T38529 D00HTY 5280363 IC50 > 10000 nM T38529 D00IQH 11677589 Ki > 5000 nM T38529 D00MZK 9911469 Ki > 10000 nM T38529 D00SOZ 44230999 IC50 = 4180 nM T38529 D01SHJ 56944705 IC50 > 10000 nM T38529 D03YAS 9824353 EC50 = 610 nM T38529 D0G6EI 9890801 EC50 = 5 nM T38529 D0K1EG 11508736 IC50 > 10000 nM T38529 D0M4TJ 44219292 Ki = 610 nM T38529 D0SP5V 49843471 IC50 = 2600 nM T38529 D0Y3LL 18376177 EC50 = 2.8 nM T38529 D0W2OT 5311035 EC50 = 33 nM T38529 D02RUO 9807448 Ki = 0.74 nM T38529 D08QHS 11296282 IC50 = 4169 nM T38529 C5Z8HC 132836 Ki = 240 nM T38529 CANV86 1498200 Ki > 8000 nM T38529 C3LM8E 1498314 Ki > 8000 nM T38529 CAV3H9 1987175 IC50 = 1600 nM T38529 C2XLU7 5311228 Ki = 1.7 nM T38529 CO7N1Z 5311239 IC50 = 4900 nM T38529 CZA41R 9808508 Ki = 14000 nM T38529 C6TA3N 9809136 Ki = 23000 nM T38529 CV24TI 9817292 Ki = 43000 nM T38529 C5WL7C 9821171 EC50 = 434 nM T38529 C5J8WP 9830442 Ki > 100000 nM T38529 CG3IS9 9830839 Ki > 10000 nM T38529 COU85R 9863804 EC50 = 595 nM T38529 C97MIQ 9865111 Ki = 940 nM T38529 C6V1BA 9872741 Ki > 100000 nM T38529 CA2I4Z 9873528 Ki = 11000 nM T38529 CKMW12 9874010 Ki = 23000 nM T38529 C38DYF 9885106 Ki = 4700 nM T38529 CF0HC5 9888589 IC50 > 10000 nM T38529 CFC8G4 9894720 Ki > 3000 nM T38529 CA5N0K 9895436 Ki > 100000 nM T38529 C7MA6V 9916766 Ki > 100000 nM T38529 CN2UX4 9938625 Ki > 100000 nM T38529 CICE70 9938626 Ki > 100000 nM T38529 C1KAC5 9938669 Ki = 22000 nM T38529 C6DQ3W 9938995 Ki > 100000 nM T38529 CWDT69 9939791 Ki = 11000 nM T38529 CWS81C 9944231 Ki = 8100 nM T38529 C4Q7RI 9953337 Ki = 8000 nM T38529 C6SGH7 9954562 Ki = 8600 nM T38529 C4UK2Q 9955802 Ki > 3000 nM T38529 C6ZM4U 9959673 Ki > 100000 nM T38529 CCD30P 9960839 Ki > 100000 nM T38529 C4Z7BL 9965922 Ki = 7300 nM T38529 C5AF0B 9975502 Ki = 134 nM T38529 CQ3GW6 10047541 IC50 = 1300 nM T38529 CQT1G4 10089562 EC50 = 23 nM T38529 CNE21V 10095268 IC50 < 3162.28 nM T38529 COR8X7 10109445 Ki = 3700 nM T38529 C6UI2Z 10111602 Ki = 750 nM T38529 CBYV78 10112486 Ki = 4100 nM T38529 C93DSI 10113454 Ki = 22000 nM T38529 C26QRM 10118889 Ki = 2000 nM T38529 C6BOW4 10144273 Ki = 16000 nM T38529 CG4YV6 10157810 Ki = 1729 nM T38529 C6W9IC 10158725 Ki = 2500 nM T38529 CM3SE6 10168694 Ki = 4900 nM T38529 C71GVU 10178073 Ki = 8100 nM T38529 CEM21G 10181606 Ki = 10000 nM T38529 C6X5CP 10202765 Ki = 29000 nM T38529 CMD93W 10204257 Ki = 6000 nM T38529 C4DLP9 10205205 Ki = 2830 nM T38529 CNT8H9 10221497 Ki = 6200 nM T38529 CP8KN7 10227492 Ki = 4600 nM T38529 CZP7B5 10229201 Ki = 2360 nM T38529 CFWB04 10247632 Ki = 802 nM T38529 C0ED9Y 10251023 IC50 > 10000 nM T38529 C47IJF 10269242 Ki = 4410 nM T38529 CQ0R3G 10270893 EC50 = 1300 nM T38529 C89CXB 10271490 Ki = 380 nM T38529 CZ21EM 10272306 Ki = 6290 nM T38529 CL7YG3 10287121 Ki > 13000 nM T38529 C40QFO 10291963 EC50 = 15 nM T38529 CK7M3E 10295421 Ki = 5690 nM T38529 C2J0PF 10298293 Ki = 5450 nM T38529 CV9QL7 10302378 Ki = 8000 nM T38529 C3C5IM 10322469 Ki > 100000 nM T38529 CB19MW 10402929 Ki = 13000 nM T38529 CT8UC2 10448293 Ki = 1850 nM T38529 C8ZB6N 10452108 Ki = 749 nM T38529 CZ1XW6 10483360 Ki = 44000 nM T38529 CI5HA0 10648334 IC50 > 10000 nM T38529 C9YQG5 10670992 IC50 = 2400 nM T38529 C7GY6X 10739351 IC50 > 10000 nM T38529 CY8IB2 10740699 IC50 > 10000 nM T38529 C12SBH 10741017 IC50 > 10000 nM T38529 CG17HE 10741197 IC50 > 10000 nM T38529 CKST02 11122314 IC50 > 10000 nM T38529 CEI08Z 11155228 Ki = 5400 nM T38529 CC8PQ2 11156167 EC50 = 60 nM T38529 CF6EO3 11210487 Ki = 8 nM T38529 CA71OC 11235004 Ki < 1995.26 nM T38529 C4S5MX 11249458 Ki > 10000 nM T38529 C70ESM 11269563 Ki = 310 nM T38529 COS4C2 11294085 EC50 = 0.67 nM T38529 C9E4SW 11294166 Ki = 390 nM T38529 CIM8K7 11328569 EC50 = 18 nM T38529 CQU62G 11337782 Ki = 220 nM T38529 C4IK7Y 11339240 Ki = 2500 nM T38529 CBP71Y 11362836 EC50 = 5.7 nM T38529 CN2TG7 11387144 Ki > 3000 nM T38529 CUWE27 11405770 Ki = 35 nM T38529 CXPO04 11408533 Ki = 230 nM T38529 CP4LS0 11440167 Ki = 75 nM T38529 CZ4K0P 11476788 Ki = 3404 nM T38529 CE2JA4 11488860 Ki = 2270 nM T38529 CW3YO5 11494768 IC50 > 10000 nM T38529 CQ6IU7 11509269 IC50 > 10000 nM T38529 CF2OM8 11539410 IC50 = 6400 nM T38529 CJ2OE0 11575201 IC50 = 1620 nM T38529 C1W2ZK 11577792 Ki = 1836 nM T38529 C7Y6XJ 11597294 Ki = 410 nM T38529 C2M8HZ 11610353 IC50 > 10000 nM T38529 CGS72I 11618662 IC50 = 3320 nM T38529 C9L5VD 11631813 IC50 > 10000 nM T38529 CMB6F9 11653874 IC50 = 6600 nM T38529 C51UDK 11667741 IC50 > 10000 nM T38529 CAL96X 11683088 IC50 = 4360 nM T38529 CW8RY9 11689895 IC50 > 10000 nM T38529 C9CM2R 11695689 IC50 > 10000 nM T38529 C3BSV4 11696697 Ki > 13000 nM T38529 CNYK74 11743212 Ki = 2300 nM T38529 CR82PA 12112238 Ki = 830 nM T38529 CX0M2W 12112239 Ki = 2900 nM T38529 C32GBT 12137443 Ki = 5100 nM T38529 CT34LO 13230981 Ki = 6680 nM T38529 CO19GA 14372497 Ki > 4600 nM T38529 C06OGJ 15486805 IC50 > 10000 nM T38529 C0L3VU 15486806 IC50 = 2500 nM T38529 CU5J6N 15491229 Ki > 100000 nM T38529 CMG0Z1 15491230 Ki > 100000 nM T38529 CWQ8B9 15551228 Ki > 100000 nM T38529 CZ87CN 15907747 Ki = 13000 nM T38529 CVEO28 15907748 Ki = 21000 nM T38529 CIS83K 15947857 Ki = 300 nM T38529 C3L0RK 15948325 Ki = 1900 nM T38529 CHBE61 15949677 IC50 > 30000 nM T38529 CRT3I2 15979081 EC50 = 0.48 nM T38529 CK4FJ8 16664733 IC50 = 32000 nM T38529 CS8M2G 18973764 Ki = 150 nM T38529 CX08BC 21198692 Ki > 40000 nM T38529 CR37AJ 21362845 Ki = 70000 nM T38529 C6UT1I 21362849 Ki = 3600 nM T38529 C4IFY8 21362851 Ki = 3700 nM T38529 C9HQN0 21362853 Ki = 2900 nM T38529 C6F8QI 21362863 Ki > 97000 nM T38529 CL5O9E 21362867 Ki = 31000 nM T38529 C58NCB 21362869 Ki > 100000 nM T38529 CHS9L6 21362879 Ki = 2900 nM T38529 CW7R1M 21362893 Ki = 2900 nM T38529 C9HD2W 21362900 Ki = 2700 nM T38529 CSUO46 21362905 Ki = 5500 nM T38529 CJ65SZ 21362910 Ki = 3500 nM T38529 CFV24G 21362912 Ki = 1800 nM T38529 C0UT6R 22008966 Ki = 6500 nM T38529 CJ4M7P 22008967 Ki = 6500 nM T38529 C9TSB7 22009003 Ki = 3900 nM T38529 C8SON3 22009004 Ki = 2415 nM T38529 CAML12 22009006 Ki = 8000 nM T38529 C5DGQ4 22009008 Ki = 8700 nM T38529 C5SJ2H 22009011 Ki = 2100 nM T38529 C3D2LR 22990263 Ki = 7500 nM T38529 CF81SW 23582412 IC50 > 10000 nM T38529 CP2S4J 23663736 Ki = 1400 nM T38529 C4VN2S 23674101 Ki = 16 nM T38529 CASU54 23696973 IC50 = 1584.89 nM T38529 C42LYP 24765153 Ki = 7323 nM T38529 CF72YI 24765671 Ki >= 785 nM T38529 C31JZP 24765672 Ki >= 2500 nM T38529 C4QX7Y 24765675 Ki >= 930 nM T38529 CL7Z9U 24765768 Ki >= 110 nM T38529 CLS5J9 24776302 IC50 > 30000 nM T38529 C4BD1L 24776306 IC50 > 30000 nM T38529 CFQA40 24952577 Ki = 16 nM T38529 CD98IN 24952580 Ki = 746 nM T38529 C81WVN 24952927 Ki = 1194 nM T38529 CZT83E 24952928 Ki > 29034 nM T38529 C8YHX3 24953283 Ki = 384 nM T38529 CZ93FO 24953285 Ki = 43 nM T38529 C17JTY 24953286 Ki = 467 nM T38529 CFT0W5 24953624 Ki > 29142 nM T38529 C42VMD 24953625 Ki = 800 nM T38529 C7B2EW 24953628 Ki = 202 nM T38529 CXQJ67 25002382 Ki >= 1291 nM T38529 CN5SH9 25003075 Ki = 8000 nM T38529 C4J2BS 25195248 IC50 = 13900 nM T38529 CR10FW 30897313 IC50 = 70 nM T38529 C6JM7A 30956824 IC50 = 200 nM T38529 CV8PE9 42484632 IC50 = 700 nM T38529 CNOF71 44138108 Ki = 3975 nM T38529 CSRV98 44157014 IC50 = 12500 nM T38529 C2O0NL 44230575 EC50 = 1.1 nM T38529 C4YFG7 44230722 EC50 = 1.6 nM T38529 C3B7MK 44230997 EC50 = 43 nM T38529 CQ13MH 44234032 Ki = 570 nM T38529 CR68BA 44250281 Ki > 10000 nM T38529 CN90FE 44269464 Ki = 3610 nM T38529 C1L0ET 44269468 Ki > 13000 nM T38529 C5KRQ4 44269486 Ki = 4050 nM T38529 CL6M2P 44269516 Ki = 3000 nM T38529 CON8R9 44269520 Ki > 13000 nM T38529 C6MBG0 44269521 Ki > 13000 nM T38529 CZ3Q1L 44269523 Ki > 13000 nM T38529 CRL61O 44269532 Ki > 13000 nM T38529 C1Z4LU 44269540 Ki > 13000 nM T38529 CM72FA 44269542 Ki > 13000 nM T38529 CN0JV2 44269543 Ki > 13000 nM T38529 C28UJH 44269544 Ki > 13000 nM T38529 CR1IY6 44269568 Ki > 13000 nM T38529 CI3C9O 44269596 Ki > 13000 nM T38529 CC0EW9 44269597 Ki > 13000 nM T38529 C6JAE2 44289921 Ki = 71000 nM T38529 CG8KT3 44289969 Ki = 41000 nM T38529 C68XKV 44289977 Ki = 68000 nM T38529 CHZ21Q 44290257 Ki > 100000 nM T38529 CO31WZ 44290262 Ki = 4200 nM T38529 COF9C2 44290263 Ki = 26000 nM T38529 C4SEW6 44290266 Ki = 6.4 nM T38529 CEVM85 44290267 Ki > 100000 nM T38529 C7RDN9 44290271 Ki = 85000 nM T38529 CN5RG9 44290272 Ki = 42000 nM T38529 CZ59QY 44290312 Ki = 32000 nM T38529 CAV76T 44290314 Ki = 58000 nM T38529 CS7RH0 44320126 Ki = 2100 nM T38529 CLR9F5 44320272 Ki = 590 nM T38529 CKYS39 44320294 Ki = 3000 nM T38529 CH6TK1 44320321 Ki = 2900 nM T38529 CYI1O0 44320373 Ki = 140 nM T38529 C0V3OA 44320388 Ki = 8600 nM T38529 C01HGT 44320405 Ki = 2500 nM T38529 CS58ZQ 44320433 Ki = 3800 nM T38529 CS52ZR 44324368 Ki = 16000 nM T38529 CM72WE 44349503 Ki = 1600 nM T38529 C9PO1Q 44349528 Ki = 4600 nM T38529 C1R7HU 44349531 Ki = 3600 nM T38529 CHO7X0 44349551 Ki = 2500 nM T38529 CLN63A 44377464 Ki = 4100 nM T38529 CJIS72 44390782 Ki = 1100 nM T38529 C43VIA 44390806 Ki = 990 nM T38529 CB8H4V 44390831 Ki = 4100 nM T38529 CWL1X4 44400355 Ki > 1000 nM T38529 C76QVA 44402710 Ki > 1000 nM T38529 CRAX23 44402824 Ki > 1000 nM T38529 CIB2W5 44419347 Ki = 5400 nM T38529 CF35LY 44419350 Ki = 940 nM T38529 CNK1X9 44419351 Ki = 1600 nM T38529 C91JXT 44419374 Ki = 860 nM T38529 CNF4W2 44419379 Ki = 860 nM T38529 CS3IW4 44419380 Ki = 2100 nM T38529 CBQ01L 44419384 Ki = 2100 nM T38529 CGS0P7 44442327 EC50 = 16 nM T38529 CF32IP 44442331 EC50 = 35 nM T38529 CZVA37 44442332 Ki = 88 nM T38529 C0IV9J 44442334 Ki = 173 nM T38529 C7HFG3 44442337 Ki = 60 nM T38529 CCV69D 44444714 Ki = 2760 nM T38529 CVH1E4 44444715 Ki = 8340 nM T38529 CZ27AC 44444716 Ki = 560 nM T38529 CQL04T 44444719 Ki = 9200 nM T38529 CE5MU6 44444720 Ki = 3070 nM T38529 CXQ5K3 44444721 Ki = 2030 nM T38529 CW60FE 44444722 EC50 = 393 nM T38529 CDBE16 44450497 Ki > 29188 nM T38529 CV8IX1 44455046 EC50 = 250 nM T38529 CRZ5K2 44455084 EC50 = 3 nM T38529 CD6B3W 44455115 EC50 = 19 nM T38529 CCY63H 44455157 Ki > 10000 nM T38529 C3DQ5V 44455158 Ki = 25000 nM T38529 C1CB7O 44455236 Ki = 54 nM T38529 CUHD74 44564571 IC50 = 4200 nM T38529 CA05LN 44564804 IC50 = 9600 nM T38529 C6XE0K 44564841 IC50 > 10000 nM T38529 CND54C 44564892 IC50 = 7680 nM T38529 C2VR6S 44564893 IC50 = 9300 nM T38529 C18GXI 44564937 IC50 > 10000 nM T38529 CZ74GB 44564990 IC50 = 10000 nM T38529 C0NF1S 44565193 IC50 > 10000 nM T38529 C07ODW 44570000 IC50 = 12261 nM T38529 CJKA53 44570666 IC50 = 2300 nM T38529 C5PT0Z 44626877 IC50 > 10000 nM T38529 CQIK27 44627395 IC50 = 4832 nM T38529 C4W1ZG 44627515 IC50 = 32921 nM T38529 C5AY6M 46220498 Ki > 8000 nM T38529 CS4F0X 46879894 IC50 = 19800 nM T38529 C2FR7X 46885690 IC50 > 20000 nM T38529 CN8D5V 46885691 IC50 > 20000 nM T38529 C9RP0X 46885735 IC50 > 20000 nM T38529 C0A2CI 46890616 Ki >= 504 nM T38529 CW52VH 46890658 Ki >= 260 nM T38529 CXQ2W0 46890659 Ki >= 580 nM T38529 CQ20RC 46890660 Ki >= 100 nM T38529 CTR7Q0 49850345 IC50 > 50118.72 nM T38529 CM06FG 50898361 Ki = 3330 nM T38529 CF1ZU9 52945294 Ki = 750 nM T38529 C4K6BH 52946883 Ki > 10000 nM T38529 CV41BH 53260154 EC50 = 4.5 nM T38529 CN4HP2 53260155 EC50 = 18 nM T38529 C87AIE 53260293 EC50 = 13 nM T38529 CWR1Z7 56665984 Ki > 13000 nM T38529 CA1DF5 57392712 IC50 > 1000 nM T38529 C96FQZ 57395059 EC50 = 5.6 nM T38529 C8RS3N 57396195 IC50 > 1000 nM T38529 CRUJ96 57399661 IC50 > 1000 nM T38529 CVLQ48 57401413 IC50 > 1000 nM T38529 CP7A2U 58905349 IC50 = 1290 nM T38529 CB1N8J 58905358 IC50 > 20000 nM T38529 C1CFM4 58905388 IC50 = 236 nM T38529 C0U1HA 59179260 Ki > 8700 nM T38529 CK7T6D 59179887 Ki > 8700 nM T38529 C4CIH9 59179917 Ki > 8700 nM T38529 CVC72I 59554822 EC50 = 2.9 nM T38529 CCXA68 59554824 EC50 = 7.4 nM T38529 C2EVC3 59554827 EC50 = 0.91 nM T38529 C8RV1N 66717319 EC50 = 75 nM T38529 C2RYV3 66717335 EC50 = 3.4 nM T38529 C7XT0A 66717343 EC50 = 5.6 nM T38529 CL4AM8 66717493 EC50 = 35 nM T38529 C2MEX7 66717697 EC50 = 307 nM T38529 C2E8BL 66717740 EC50 = 2 nM T38529 CNUA34 66857670 EC50 = 21 nM T38529 C1WA3L 66857738 EC50 = 3700 nM T38529 C1C3AF 66857975 EC50 = 92 nM T38529 CUIV04 66857988 EC50 = 2.1 nM T38529 CB56OD 66858036 EC50 = 3400 nM T38529 CU5V8I 66858111 EC50 = 160 nM T38529 CB2J4V 66978356 EC50 = 0.086 nM T38529 C4FHO2 67082722 EC50 = 6.8 nM T38529 CGQA79 67082748 EC50 = 0.37 nM T38529 CVM9Q1 68503758 IC50 > 10000 nM T38529 CA15ND 68505312 IC50 > 10000 nM T38529 C0US2T 68505327 IC50 = 7400 nM T38529 CX8W7F 68508048 IC50 > 10000 nM T38529 C5NZO0 68747479 EC50 > 10000 nM T38529 CJ7AY6 69753740 EC50 = 8900 nM T38529 CU7O4C 70815427 EC50 = 19 nM T38529 C3POW5 70815457 EC50 = 6.1 nM T38529 CNU70Y 70815480 EC50 = 2.8 nM T38529 C69IFJ 70815631 EC50 = 2.7 nM T38529 C4BYT6 70815856 EC50 = 45 nM T38529 CJD1M3 70815950 EC50 = 119 nM T38529 CB16FR 70816051 EC50 = 4.4 nM T38529 C4UQI3 70816091 EC50 = 2.6 nM T38529 CLKZ81 70816117 EC50 = 2.7 nM T38529 C9UJ8Q 70816208 EC50 = 4.3 nM T38529 CQD9Y0 70816226 EC50 = 109 nM T38529 C01YOJ 71452690 Ki = 63 nM T38529 CQ5E0J 71455094 Ki = 10810 nM T38529 COK0V6 71458757 Ki = 2943 nM T38529 C74PUE 71462285 Ki = 4264 nM T38529 C8XJ0I 71733818 IC50 > 10000 nM T38529 CXC78L 71733909 IC50 > 10000 nM T38529 C7B5XE 71733910 IC50 = 2700 nM T38529 CQ21ZD 71733911 IC50 > 10000 nM T38529 CZG0S2 71733912 IC50 = 9500 nM T38529 C4G2UR 72695027 Ki = 1210 nM T38529 CDFO42 72695136 Ki > 18900 nM T38529 CX6T7A 72706947 EC50 > 10000 nM T38529 C6PLC5 72722131 Ki = 4971 nM T38529 CU39ZO 72950089 Ki = 329 nM T38529 CWTO83 91810751 Ki > 18900 nM T38529 CR4DE7 118175009 Ki = 2800 nM T38529 CSJ4A9 118352160 EC50 = 0.69 nM T38529 CE6L8I 118352177 EC50 = 23 nM T38529 C8PKA7 118352211 EC50 = 13 nM T38529 CUZX68 118352215 EC50 = 2.9 nM T38529 CPS7M4 118352285 EC50 = 2.2 nM T38529 CR5Y0C 118756024 IC50 = 14000 nM T38529 CP85OZ 122180249 IC50 = 20 nM T38529 CDOY04 122180250 IC50 = 200 nM T38529 C63OBS 122180251 IC50 = 1500 nM T38529 CG1BK6 122180252 IC50 = 200 nM T38529 CG8A9X 122180253 IC50 = 10000 nM T38529 CP4J1U 122180254 IC50 = 30000 nM T38529 C9F7RC 122180255 IC50 = 30000 nM T38529 C8K0UY 122180256 IC50 = 1800 nM T38529 CEL3P1 122180257 IC50 = 600 nM T38529 C40IXF 122180258 IC50 = 600 nM T38529 CHPO27 122180259 IC50 = 100 nM T38529 C0UY6A 122180260 IC50 = 30000 nM T38529 C76IFQ 122180261 IC50 = 100 nM T38529 CXD45K 122180262 IC50 > 30000 nM T38529 CTEI17 122180263 IC50 = 2800 nM T38529 CDZH05 122180264 IC50 = 15000 nM T38529 CHSK65 122180265 IC50 = 300 nM T38529 C3SM2Q 122180266 IC50 > 30000 nM T38529 CRW2O5 122180267 IC50 = 13000 nM T38529 CS65YL 122180268 IC50 > 30000 nM T38529 C5MR2O 122180269 IC50 = 12000 nM T38529 CRB2Y5 122180270 IC50 = 700 nM T38529 CA45NB 122180271 IC50 = 10000 nM T38529 CW75AL 122180272 IC50 = 400 nM T38529 CK1C9Y 122180273 IC50 = 15000 nM T38529 CK6WS2 122180274 IC50 = 300 nM T38529 CY0LE2 122180275 IC50 = 2700 nM T38529 C8X1OV 122180276 IC50 = 1100 nM T38529 CC2E6B 122180277 IC50 = 60 nM T38529 C9T4YN 122180278 IC50 = 400 nM T38529 C0FN7C 122180279 IC50 = 700 nM T38529 CKY4Q7 122180280 IC50 = 4000 nM T38529 CRIL37 122180281 IC50 = 5600 nM T38529 CZNI51 122180282 IC50 = 100 nM T38529 CF4S5Z 122180283 IC50 = 40 nM T38529 CGBT75 122180284 IC50 = 30 nM T38529 CVAJ62 122180285 IC50 = 1100 nM T38529 CE8A9T 122180286 IC50 = 3800 nM T38529 CQZF36 122180287 IC50 > 30000 nM T38529 CHLO48 122180288 IC50 = 200 nM T38529 C7Z3HU 122180289 IC50 = 80 nM T38529 CSFB97 122180290 IC50 = 1600 nM T38529 CL63VX 122180291 IC50 = 6000 nM T38529 C4JUT7 122180292 IC50 = 4000 nM T38529 C7PFK8 122180293 IC50 = 13000 nM T38529 CN7R3X 122180294 IC50 > 30000 nM T38529 C2NG1J 122180295 IC50 = 20 nM T38529 CT2K3E 126495360 EC50 = 27 nM T38529 C8ZRJ0 126495398 EC50 = 10 nM T38529 CD61VL 126495400 EC50 = 0.21 nM T38529 CW79RH 126495420 EC50 = 28 nM T38529 CVP0M7 126495424 EC50 = 3.6 nM T38529 C8SRZ5 126495427 EC50 = 114 nM T38529 CD72CT 126495432 EC50 = 55 nM T38529 CN72WL 126495463 EC50 = 1.4 nM T38529 CV1A6C 126495491 EC50 = 13 nM T38529 CYP3E5 126495507 EC50 = 11 nM T38529 C2N7XJ 127026652 EC50 = 29 nM T38529 C8KYB6 127026952 EC50 = 2 nM T38529 C8VI4F 127026953 EC50 = 1.8 nM T38529 C5M4LU 127026954 EC50 = 3.9 nM T38529 COT2I4 127026955 EC50 = 0.17 nM T38529 CVJ30Z 127026956 EC50 = 0.2 nM T38529 CX5WL8 127027874 EC50 = 0.9 nM T38529 CEN4D9 127027875 EC50 = 3.9 nM T38529 CAT1I9 127027876 EC50 = 0.11 nM T38529 C94DAB 127027877 EC50 = 0.57 nM T38529 C3BR0Q 127028169 EC50 = 0.68 nM T38529 CX9M6D 127029402 EC50 = 15 nM T38529 CWXR72 127029417 Ki > 50000 nM T38529 CW1O4F 127029692 EC50 = 0.14 nM T38529 C0UJ5N 127037150 EC50 = 0.39 nM T38529 CJAQ90 127047381 Ki > 50000 nM T38529 CBCQ64 127047601 Ki > 10000 nM T38529 CUHN85 127050450 EC50 = 5.4 nM T38529 CZP04R 127050451 EC50 = 14 nM T38529 C5H1WU 127050452 EC50 = 13 nM T38529 CJ96UM 127050766 EC50 = 7 nM T38529 C7Q9AE 127051062 EC50 = 3.3 nM T38529 C3S1ZJ 127051063 EC50 = 0.5 nM T38529 C6FQX2 127051064 EC50 = 23 nM T38529 CP4KT3 127051656 EC50 = 0.9 nM T38529 C62OMX 127052577 EC50 = 6.5 nM T38529 CTR62O 127052613 EC50 = 7.9 nM T38529 CGZR45 127052614 EC50 = 3.9 nM T38529 COVY75 127052615 EC50 = 3.8 nM T38529 CA8QC3 141730897 IC50 > 10000 nM T38529 C2P9GV 141730900 IC50 > 10000 nM T38529 CK6E7L 141730914 IC50 > 10000 nM T38529 C7B5WG 141730916 IC50 > 10000 nM T38529 C62DUY 141730923 IC50 > 10000 nM T38529 CSXG54 145965248 EC50 = 31 nM T38529 CIS1V8 145966519 EC50 = 2 nM T38529 C54SAN 145971909 EC50 = 0.068 nM T38529 CGV2E8 145977227 EC50 = 1.1 nM T38529 CLVI73 145978309 EC50 = 0.11 nM T38529 CDN70S 146014480 IC50 > 10000 nM T38529 CM9QA1 155516303 Ki = 15 nM T38529 COER95 155520370 Ki = 433 nM T38529 CY9K4V 155521506 EC50 = 83 nM T38529 CZ10RG 155522808 IC50 > 10000 nM T38529 C3XJR1 155527946 EC50 = 620 nM T38529 C7UY3Q 155529786 IC50 > 10000 nM T38529 C7ZI9E 155532079 EC50 = 29 nM T38529 C2KIH7 155532594 EC50 > 1000 nM T38529 CP43IA 155539237 EC50 = 649 nM T38529 C9VA4G 155541718 EC50 = 283 nM T38529 CM8FU4 155542680 EC50 = 360 nM T38529 C95YVD 155544327 EC50 > 1000 nM T38529 CJM86N 155550015 EC50 = 118 nM T38529 C82RVN 155554217 IC50 > 10000 nM T38529 CWU1C5 155556219 EC50 = 91 nM T38529 C71RSA 155566381 EC50 > 1000 nM T38529 C4TR5H 155569438 EC50 > 1000 nM T38529 D02LXJ 9813912 Ki = 1400 nM T38529 D02MXT 24952929 Ki = 5900 nM T38529 D02SAD 44419388 Ki = 2500 nM T38529 D03OYD 5311240 IC50 = 6700 nM T38529 D07JMB 44289922 Ki = 1459 nM T38529 D07UDT 15551229 Ki > 50000 nM T38529 D08MNO 25886893 EC50 = 32 nM T38529 D0H5TU 11524454 IC50 = 709 nM T38529 D0J9PG 119461 Ki = 1150 nM T38529 D0O9ES 5311053 IC50 = 3700 nM T38529 D0QH5C 230826 Ki = 3000 nM T38529 D0S2LO 9864831 Ki > 13000 nM T38529 D0ST1M 673766 EC50 = 7800 nM T38529 D0TA0L 23685469 Ki > 1000 nM T38529 D0Y1IF 23664784 Ki > 1000 nM T38529 D0Z3XJ 9817405 Ki = 12000 nM T82028 D0I0RJ 16231 IC50 = 66730 nM T82028 D0N8QQ 151172 IC50 = 680 nM T82028 D0V9RU 6433092 IC50 = 140 nM T82028 COE28J 7220 IC50 = 192680 nM T82028 CN6X7A 25902 IC50 = 97100 nM T82028 CEM5Y1 27939 IC50 = 86480 nM T82028 CCSR93 85498 IC50 = 177000 nM T82028 C1NS4W 178019 IC50 = 1200 nM T82028 C0S8TR 521212 IC50 = 72510 nM T82028 C64ZIJ 570059 IC50 = 51570 nM T82028 C96AKN 590090 IC50 = 355000 nM T82028 CH4S3X 594606 IC50 = 65140 nM T82028 CM87JK 750248 IC50 = 50890 nM T82028 C8GBK3 1380969 IC50 = 49950 nM T82028 CKB14W 3343351 IC50 = 101120 nM T82028 C1I5AN 3477267 IC50 = 115250 nM T82028 CA7EP3 3708772 IC50 = 63470 nM T82028 C91AEO 3754503 IC50 = 72380 nM T82028 C2WCD8 3789956 IC50 = 156540 nM T82028 C54DAY 3797398 IC50 = 154670 nM T82028 CI12GP 4202453 IC50 = 60590 nM T82028 C8C0BP 4311536 IC50 = 135000 nM T82028 C2PE6M 4359223 IC50 = 59230 nM T82028 CZUA02 4401906 IC50 = 68110 nM T82028 C4Y2QR 5243938 IC50 = 69750 nM T82028 C6H1QB 5244322 IC50 = 191230 nM T82028 C6H4DT 6433110 IC50 = 59 nM T82028 C5X3SL 9796199 IC50 = 180 nM T82028 CZ39AI 9816854 IC50 = 350 nM T82028 C1K7TP 9816861 IC50 = 3800 nM T82028 CZJ48L 9817020 IC50 = 39 nM T82028 C2XM5R 9818623 IC50 = 3600 nM T82028 C0F2HT 9838628 IC50 = 4000 nM T82028 CNM7Q3 9860589 IC50 = 2600 nM T82028 C74JKE 9868115 IC50 = 28 nM T82028 CTB2S9 9881852 IC50 = 11000 nM T82028 CWC0M2 9925502 IC50 = 9 nM T82028 C9T7JD 10131262 IC50 > 30000 nM T82028 CKG2R4 10336075 IC50 = 160 nM T82028 C15KVI 10860947 IC50 = 540 nM T82028 CA2S4J 10862369 IC50 = 17 nM T82028 C64FPC 10862562 IC50 = 5 nM T82028 C4IE9O 10893528 IC50 = 2900 nM T82028 C6D5YB 10925702 IC50 = 1600 nM T82028 C9YT3D 10948894 IC50 = 14 nM T82028 C9CZI4 10958084 IC50 = 3500 nM T82028 CXV1U9 10960633 IC50 = 6 nM T82028 CPUN94 11014654 IC50 = 5 nM T82028 CO8M2C 11057914 IC50 = 32 nM T82028 CT7LM1 11078662 IC50 = 280 nM T82028 CU0X3P 11078949 IC50 = 1600 nM T82028 C3AZW8 11086037 IC50 = 120 nM T82028 CI8E9X 11090105 IC50 = 12 nM T82028 CL58JI 11090964 IC50 = 90 nM T82028 CFE10D 11091487 IC50 = 3 nM T82028 CQ87FM 11110736 IC50 = 69 nM T82028 CK2W0B 11122007 IC50 > 30000 nM T82028 CMTK82 11132107 IC50 > 30000 nM T82028 C0GZ2L 11149755 IC50 = 1300 nM T82028 C1SN6I 11149756 IC50 > 30000 nM T82028 C0TYL7 11151941 IC50 > 30000 nM T82028 CXIP24 11153069 IC50 = 140 nM T82028 CV7L8T 11153588 IC50 = 2000 nM T82028 CW02VL 11161203 IC50 = 3700 nM T82028 CT70QA 11196783 IC50 > 30000 nM T82028 C51HEB 11207657 IC50 = 7400 nM T82028 COIW49 11230628 IC50 = 650 nM T82028 CM1UQ6 11230686 IC50 > 30000 nM T82028 CJD02R 11242380 IC50 = 2300 nM T82028 C2N5YP 11242502 IC50 = 27000 nM T82028 CMC48K 11256959 IC50 = 15000 nM T82028 C5Q2PW 11276980 IC50 = 1700 nM T82028 CRE7O8 11293275 IC50 > 30000 nM T82028 C8J5WX 11299864 IC50 = 3000 nM T82028 CD5OI7 11300040 IC50 = 750 nM T82028 C59AVD 11300292 IC50 > 30000 nM T82028 C5P9MV 11311839 IC50 = 2600 nM T82028 C7PRX3 11312289 IC50 > 30000 nM T82028 CD2ZN5 11313895 IC50 = 3500 nM T82028 CSU2E1 11323024 IC50 = 1100 nM T82028 CWLM79 11324276 IC50 = 140 nM T82028 CYN0I7 11326836 IC50 = 9400 nM T82028 C9XRS8 11334583 IC50 = 7900 nM T82028 C5N2FX 11356966 IC50 > 30000 nM T82028 CZ1YQ8 11358162 IC50 = 2400 nM T82028 CTPY63 11368995 IC50 = 230 nM T82028 CC6X4U 11391762 IC50 = 480 nM T82028 C7U2GX 11393090 IC50 = 130 nM T82028 C5IME4 11403628 IC50 = 81 nM T82028 CF08HG 11413943 IC50 = 39000 nM T82028 C51UGZ 11425071 IC50 = 20000 nM T82028 CJ1IU7 11447917 IC50 > 30000 nM T82028 CA8GZ5 11447995 IC50 = 2400 nM T82028 CKH05R 11449112 IC50 = 4400 nM T82028 C1K7OE 11460688 IC50 > 30000 nM T82028 C2QN1E 11461388 IC50 = 1100 nM T82028 C02ANQ 11461861 IC50 = 93 nM T82028 C1XY7E 11472035 IC50 = 730 nM T82028 CP5G9N 11482285 IC50 = 4400 nM T82028 CU0N3Z 11483373 IC50 = 120 nM T82028 CH80ZS 11495212 IC50 = 11000 nM T82028 CN6RB2 11495616 IC50 = 5100 nM T82028 CYHB68 11495618 IC50 = 8900 nM T82028 CD1F8T 11500855 IC50 = 480 nM T82028 CS6J2M 11502339 IC50 = 3400 nM T82028 CD1B2P 11508455 IC50 = 3400 nM T82028 CTE98F 11515637 IC50 = 2000 nM T82028 CT71CE 11545926 IC50 = 7700 nM T82028 C7ZO1L 11558719 IC50 = 12000 nM T82028 CL38RQ 11560573 IC50 = 3900 nM T82028 CAR06Z 11560834 IC50 = 11000 nM T82028 CP7GC9 11561645 IC50 = 4400 nM T82028 CQ51SI 11581271 IC50 = 2300 nM T82028 CVH9O4 11581912 IC50 = 8400 nM T82028 CIOA15 11603377 IC50 = 400 nM T82028 CY54ES 11610895 IC50 = 200 nM T82028 CUPH75 11611606 IC50 = 4200 nM T82028 C6KDQ9 11617077 IC50 = 310 nM T82028 C9JBN5 11617121 IC50 = 270 nM T82028 C1DL0P 11631799 IC50 = 850 nM T82028 C2NB3H 11640819 IC50 = 2500 nM T82028 CA4TE2 11667124 IC50 = 1700 nM T82028 CD8P3F 11668682 IC50 = 5600 nM T82028 CTY8D3 11676563 IC50 = 170 nM T82028 CS5YM3 11688868 IC50 = 200 nM T82028 C1SC4M 11689961 IC50 > 30000 nM T82028 C1TS7W 11695621 IC50 > 30000 nM T82028 C3UHY1 11711576 IC50 > 30000 nM T82028 CGZR47 11719550 IC50 = 680 nM T82028 CY20DB 11731793 IC50 = 40 nM T82028 C3KY0B 11737171 IC50 = 1300 nM T82028 CNIE21 11737807 IC50 > 30000 nM T82028 CED97O 11738059 IC50 = 1700 nM T82028 C1JOU2 11783118 IC50 = 980 nM T82028 C6LT8E 11818165 IC50 > 30000 nM T82028 CV53MT 16046241 IC50 = 6.5 nM T82028 CU54NY 16664857 IC50 = 10 nM T82028 C5J8PF 20778950 IC50 = 5.4 nM T82028 CX6M0K 20779024 IC50 = 27 nM T82028 CR36ZY 20779025 IC50 = 250 nM T82028 C2GCS3 20779027 IC50 = 1000 nM T82028 CV1A9H 20779028 IC50 = 8600 nM T82028 CER60I 20779043 IC50 = 580 nM T82028 C4SO6L 20779044 IC50 = 820 nM T82028 CL6ZW5 20779070 IC50 = 61 nM T82028 C0JKT1 20779071 IC50 = 940 nM T82028 C0S4TG 20779084 IC50 = 15 nM T82028 COP2K4 20779089 IC50 = 41 nM T82028 CGQC71 20779094 IC50 = 61 nM T82028 CU3FS7 20779096 IC50 = 350 nM T82028 CFH7J1 20779100 IC50 = 350 nM T82028 CE3S6D 20779101 IC50 = 7.4 nM T82028 C2WP3S 20779104 IC50 = 21 nM T82028 C5GKC4 20779158 IC50 = 1900 nM T82028 CF81XE 22267617 IC50 = 830 nM T82028 CZ3GS5 22267755 IC50 = 860 nM T82028 C74WHI 24905408 IC50 = 240 nM T82028 C4VZ8G 25011757 IC50 = 12000 nM T82028 C9QU5B 25011762 IC50 = 2400 nM T82028 CB62PD 25011769 IC50 = 6600 nM T82028 CO1Q4K 25011771 IC50 > 30000 nM T82028 C3E9SM 25011773 IC50 > 30000 nM T82028 C32UAL 25011775 IC50 = 1100 nM T82028 CUS8O9 25011777 IC50 > 30000 nM T82028 C1Q6BK 25011779 IC50 = 4100 nM T82028 CL7D0P 25011781 IC50 > 30000 nM T82028 C0ZBP6 25011783 IC50 > 30000 nM T82028 COB7D4 25011785 IC50 = 5000 nM T82028 C7V2DI 25011787 IC50 = 7200 nM T82028 CE46RD 25011789 IC50 = 3000 nM T82028 C0CV2L 25011793 IC50 = 12000 nM T82028 C68NMX 25011795 IC50 = 4500 nM T82028 C8F9RK 25011797 IC50 = 2700 nM T82028 CX1ZP9 25011799 IC50 = 3100 nM T82028 CU96QY 25014484 IC50 = 1400 nM T82028 CMB52E 25014485 IC50 = 4500 nM T82028 CR40VE 25014487 IC50 > 30000 nM T82028 CR5L2Q 25014489 IC50 = 500 nM T82028 CZ8F0A 25014491 IC50 = 100 nM T82028 C91PSZ 25014492 IC50 = 520 nM T82028 CGXM81 25103539 IC50 = 8200 nM T82028 C3HVY7 25103541 IC50 = 6600 nM T82028 CXU7E9 25103544 IC50 = 220 nM T82028 C4DVI7 25103670 IC50 = 7100 nM T82028 CH0M9U 25103675 IC50 = 4200 nM T82028 CQP75S 25103678 IC50 = 3300 nM T82028 CJQ15I 25103792 IC50 = 2800 nM T82028 CIQP35 25103794 IC50 = 1700 nM T82028 CBK01W 25103795 IC50 > 30000 nM T82028 CJB0R8 25103797 IC50 = 72 nM T82028 C92NYG 25103798 IC50 = 890 nM T82028 C9HXP6 25125800 IC50 = 680 nM T82028 CJ6VT4 25125801 IC50 = 15 nM T82028 CFC05W 44295851 IC50 = 30000 nM T82028 CAB0O7 44295852 IC50 = 8000 nM T82028 CRA9P6 44295900 IC50 = 10000 nM T82028 CCMN05 44295928 IC50 = 750 nM T82028 C3CE7M 44295947 IC50 = 950 nM T82028 C7QU2M 44295989 IC50 > 30000 nM T82028 C59QXI 44296003 IC50 > 30000 nM T82028 CC4AG5 44296047 IC50 > 30000 nM T82028 CCK53E 44296072 IC50 = 4850 nM T82028 CDK41P 44296073 IC50 = 8 nM T82028 C2U6DY 44402707 IC50 = 2500 nM T82028 C9YI7E 44402727 IC50 = 8600 nM T82028 C5AWL2 44416039 IC50 = 4.6 nM T82028 CAU9G6 44416040 IC50 = 87 nM T82028 CBSG85 44416089 IC50 = 11000 nM T82028 C27GTW 44416155 IC50 = 520 nM T82028 CW4NY8 44432194 IC50 = 2300 nM T82028 C3KV0O 44432195 IC50 = 1200 nM T82028 C68JMG 44432196 IC50 = 240 nM T82028 CZ13GW 44432197 IC50 = 150 nM T82028 C2M5AF 44432200 IC50 = 150 nM T82028 CP35LO 44432202 IC50 = 770 nM T82028 CZAF10 44432205 IC50 = 410 nM T82028 CJ2U4M 44432209 IC50 = 8 nM T82028 C4Q1YC 44432211 IC50 = 72 nM T82028 CP6X1S 44432216 IC50 = 120 nM T82028 CFQ74A 44432218 IC50 = 24 nM T82028 CG83EC 44432219 IC50 = 130 nM T82028 CKV7H2 44432224 IC50 = 120 nM T82028 C60CBD 44432225 IC50 = 120 nM T82028 CVH6E5 44432226 IC50 = 9 nM T82028 CK34SU 44432227 IC50 = 12 nM T82028 C5H4CF 44432228 IC50 = 14000 nM T82028 C3MY0G 44432229 IC50 = 14000 nM T82028 C1KH4O 44432230 IC50 = 6200 nM T82028 CX6N7J 44432231 IC50 = 4500 nM T82028 CZI94D 44432232 IC50 > 30000 nM T82028 C3P4BW 44432233 IC50 > 30000 nM T82028 C4POI8 44432234 IC50 > 30000 nM T82028 CM8D5L 44432235 IC50 = 33000 nM T82028 C5WAO4 44432236 IC50 = 820 nM T82028 C9RX5F 44432237 IC50 = 820 nM T82028 CN68HU 44432238 IC50 = 96 nM T82028 CG1UT5 44432239 IC50 = 5100 nM T82028 CE2R5P 44432240 IC50 = 0.48 nM T82028 C6DQ1G 44432241 IC50 = 16000 nM T82028 C3S5RP 44432242 IC50 = 480 nM T82028 CO3B7K 44432243 IC50 = 3000 nM T82028 C5AZ8M 44432244 IC50 = 24 nM T82028 C7E3YR 44432245 IC50 = 16 nM T82028 C6QP1W 44432246 IC50 = 230 nM T82028 CQ6F8I 44432247 IC50 = 5600 nM T82028 C4F5KT 44564852 IC50 = 2100 nM T82028 CZM95D 44565001 IC50 = 800 nM T82028 C9GWF1 44609645 IC50 = 5 nM T82028 CX9H3K 44610103 IC50 = 52 nM T82028 CXQ19C 44610104 IC50 = 16 nM T82028 CXB2Q6 51031001 IC50 = 31 nM T82028 CJBQ04 58269501 IC50 = 21 nM T82028 CI45ZP 58269513 IC50 = 68 nM T82028 CK10DA 58269516 IC50 = 184 nM T82028 CV9FC4 58269518 IC50 = 25 nM T82028 CLVM72 58269522 IC50 = 47 nM T82028 CM1GN4 58269523 IC50 = 14 nM T82028 CFTY53 58269531 IC50 = 58 nM T82028 C2MTF0 58269538 IC50 = 22 nM T82028 CW62SY 58269539 IC50 = 169 nM T82028 C12FCO 58269548 IC50 = 36 nM T82028 CR1PE7 58269551 IC50 = 320 nM T82028 CAY0H7 58269562 IC50 = 50 nM T82028 CN13SI 58269563 IC50 = 15 nM T82028 CS1KM2 58269577 IC50 = 306 nM T82028 C3F5KA 58269585 IC50 = 4705 nM T82028 CPQ0Z4 58269588 IC50 = 10 nM T82028 CWR57J 58269592 IC50 = 498 nM T82028 C8A3JQ 58269598 IC50 = 28 nM T82028 CD18IU 58269609 IC50 = 35 nM T82028 CFPH18 58269614 IC50 = 45 nM T82028 CQV75S 58269620 IC50 = 36 nM T82028 CF1TI9 58269622 IC50 = 33 nM T82028 C26OPT 58269625 IC50 = 18 nM T82028 C8ILS3 58269629 IC50 = 72 nM T82028 CQLA54 58269634 IC50 = 266 nM T82028 CL25UN 58269650 IC50 = 102 nM T82028 CFB1X6 58269652 IC50 = 50 nM T82028 C5VFQ7 58269655 IC50 = 24 nM T82028 CH4LO0 58269661 IC50 = 64 nM T82028 CQ63WZ 58269663 IC50 = 62 nM T82028 CL14UD 58269664 IC50 = 385 nM T82028 C2PYB1 58269668 IC50 = 14 nM T82028 CI3P0D 58269670 IC50 = 79 nM T82028 C5RF8T 58269685 IC50 = 61 nM T82028 C4OS3J 58269689 IC50 = 18 nM T82028 C3CFB8 58269691 IC50 = 11 nM T82028 C9K7YW 58269713 IC50 = 108 nM T82028 CDC14E 58269716 IC50 = 29 nM T82028 CO1DG9 58269724 IC50 = 15 nM T82028 CZ3FD4 58269726 IC50 = 19 nM T82028 CSV82P 58269734 IC50 = 27 nM T82028 CZFC05 58269741 IC50 = 15 nM T82028 CR4LZ1 66559503 IC50 = 30 nM T82028 CD2UK7 66559583 IC50 = 172 nM T82028 CO72XW 66560392 IC50 = 36 nM T82028 C60LQZ 66560393 IC50 = 41 nM T82028 CJ7YU6 134137115 IC50 > 100000 nM T82028 D01ZIP 11172909 IC50 = 1400 nM T82028 D06AKW 11390872 IC50 = 6000 nM T82028 D08BDI 11218749 IC50 = 340 nM T82028 D09ZSK 11470226 IC50 = 3100 nM T82028 D0D3OX 11349219 IC50 = 2300 nM T82028 D0V5NZ 1795 IC50 = 800 nM T96144 D01DBQ 452548 IC50 = 62700 nM T96144 D02PMO 60700 IC50 = 480 nM T96144 D07VLY 31703 IC50 = 1200 nM T96144 D0B7EB 36462 EC50 = 810 nM T96144 D0G9YH 2179 EC50 = 720 nM T96144 D0O1WX 2764 EC50 = 30 nM T96144 D0Q0PR 54675769 IC50 > 400 ug.mL-1 T96144 D0I1DW 9808998 EC50 > 50000 nM T96144 D03GQC 122796 EC50 = 340000 nM T96144 D0B3CT 9928668 EC50 > 50000 nM T96144 D0G6XC 3035776 EC50 = 3000 nM T96144 D0Q1RC 10474948 IC50 = 510 nM T96144 D0S0XS 9909677 EC50 > 480000 nM T96144 C4DTF0 6665 IC50 > 500000 nM T96144 CA4IO8 115150 IC50 = 13900 nM T96144 CDN9I7 119367 EC50 = 1200 nM T96144 CI5K0N 129581 EC50 = 9400 nM T96144 CY16ER 130078 EC50 = 7600 nM T96144 C2P6EC 372648 EC50 = 1700 nM T96144 CBE0Z6 391373 IC50 = 9000 nM T96144 C2WA5T 462428 IC50 = 500 nM T96144 CQP57I 9802791 IC50 > 500000 nM T96144 CU6NE0 9866430 EC50 = 20000 nM T96144 CTE0G7 9868285 EC50 = 96 nM T96144 CTW52L 9886271 EC50 > 260000 nM T96144 C71WVO 9887873 IC50 = 9 nM T96144 COH21F 9888201 EC50 = 980 nM T96144 CKX02G 9909579 IC50 = 150 nM T96144 CL9BG2 9910942 EC50 = 2600 nM T96144 C9RNT6 9933099 EC50 > 220000 nM T96144 C9T4OU 9954434 IC50 = 240 nM T96144 C3Q7PU 9976692 IC50 = 20000 nM T96144 C75MXR 9979116 IC50 < 1000 nM T96144 CS1Q4A 9997468 IC50 = 25000 nM T96144 CC0EN3 9998338 EC50 = 90000 nM T96144 CN36HE 10004256 IC50 = 500 nM T96144 CQ41UP 10017730 IC50 = 25000 nM T96144 C70AOB 10045694 IC50 = 20000 nM T96144 C1GX3K 10049918 EC50 > 210000 nM T96144 C1S6ZO 10053929 EC50 > 50000 nM T96144 CP62NU 10066958 IC50 = 20000 nM T96144 CWFA38 10068583 EC50 > 260000 nM T96144 C7GBZ0 10094097 IC50 = 54 nM T96144 CFNO13 10248698 IC50 = 116 nM T96144 CI4LZ7 10252167 IC50 = 490 nM T96144 CKC38F 10255039 IC50 = 2970 nM T96144 C2WZ4U 10322576 IC50 = 20 nM T96144 CE7ZT9 10334120 IC50 = 28500 nM T96144 CV47BO 10341523 EC50 > 240000 nM T96144 C5JW1M 10342927 IC50 = 63 nM T96144 C4LHU9 10346280 IC50 < 1000 nM T96144 C21JVU 10362559 EC50 = 510000 nM T96144 C9VP3J 10364521 IC50 = 20000 nM T96144 CHT85I 10365443 IC50 = 550 nM T96144 C7JS5A 10384589 IC50 = 3.2 ug.mL-1 T96144 C7NGB6 10385895 IC50 = 45 nM T96144 C9B2AU 10414142 IC50 > 100000 nM T96144 C4EM6S 10426517 EC50 = 17000 nM T96144 CYAV26 10434467 IC50 > 400 ug.mL-1 T96144 C8AZ0G 10447591 IC50 > 100000 nM T96144 C3CL8F 10452276 IC50 = 40500 nM T96144 CEF6X7 10453745 IC50 = 50000 nM T96144 C5ND4G 10456245 EC50 = 550 nM T96144 CBQ3U1 10471090 IC50 > 100000 nM T96144 CI1NW7 10473525 IC50 = 6.4 ug.mL-1 T96144 CVI31H 10478426 EC50 > 220000 nM T96144 C9OGN1 10478620 IC50 = 34.21 ug.mL-1 T96144 CA3IR4 10501735 EC50 > 240000 nM T96144 CTS76B 10521963 EC50 > 250000 nM T96144 CIU90P 10547820 EC50 > 260000 nM T96144 CULK80 10555744 IC50 = 15 ug.mL-1 T96144 CQ6CY9 10576072 EC50 > 210000 nM T96144 CRB5F3 10598750 EC50 > 230000 nM T96144 CKQF84 10618700 EC50 = 150000 nM T96144 CY51UZ 10618929 EC50 > 220000 nM T96144 C7WCR1 10622496 EC50 = 1600 nM T96144 C23LHO 10646103 EC50 = 330 nM T96144 C5O4HY 10647065 IC50 > 500000 nM T96144 CCDH96 10668643 EC50 > 500000 nM T96144 CV65XC 10671228 EC50 = 500 nM T96144 COD25P 10765128 IC50 = 770 nM T96144 C6IJT5 10765129 IC50 = 770 nM T96144 C7T2KQ 10785350 EC50 > 270000 nM T96144 CTB9F2 10812579 IC50 = 9600 nM T96144 CLN38G 10916071 IC50 = 38000 nM T96144 CMK4D3 10937930 IC50 > 150000 nM T96144 CCG3Y1 11456414 IC50 = 60 ug.mL-1 T96144 CV4WH1 11483874 IC50 = 25000 nM T96144 CECV23 11604842 IC50 > 400 ug.mL-1 T96144 CW92BH 11740959 EC50 = 13000 nM T96144 CE86RH 11794504 EC50 = 10000 nM T96144 CL3R0U 11796931 IC50 = 1840 nM T96144 C5U9SC 11796932 IC50 = 640 nM T96144 CR5UV0 13009345 EC50 > 50000 nM T96144 CN3R8Q 13009346 EC50 > 50000 nM T96144 CEW95R 13009351 EC50 > 50000 nM T96144 C0DCE1 13009352 EC50 > 50000 nM T96144 C53JGS 13009354 EC50 > 50000 nM T96144 CU9G8A 13009355 EC50 > 50000 nM T96144 CEH9V5 13727605 IC50 > 200 ug.mL-1 T96144 C45OUJ 13795334 IC50 = 200 ug.mL-1 T96144 C9VL7U 13958508 EC50 > 570000 nM T96144 CNG93D 14501361 EC50 = 50000 nM T96144 CS68HY 14501368 EC50 = 31000 nM T96144 C7NQV6 14501369 EC50 > 540000 nM T96144 CP8X7L 14501400 EC50 = 420000 nM T96144 CMZO19 14969588 EC50 > 430000 nM T96144 CMO9S8 14969591 EC50 = 110000 nM T96144 C48MTL 14969592 EC50 > 530000 nM T96144 C3HCS1 14969593 EC50 > 300000 nM T96144 CL4M9Z 14969595 EC50 > 260000 nM T96144 CM7FQ1 14969596 EC50 > 220000 nM T96144 CO0Z6E 14969597 EC50 = 16000 nM T96144 CN8MY1 14969598 EC50 > 240000 nM T96144 C3NVB7 14969599 EC50 = 6200 nM T96144 C5GD1U 14969600 EC50 > 420000 nM T96144 CW9JF6 14969601 EC50 = 16000 nM T96144 C96PWB 14969602 EC50 = 17000 nM T96144 CER9B0 14969603 EC50 = 53000 nM T96144 CD3NI6 14969604 EC50 = 52000 nM T96144 CN0QF6 15224739 EC50 = 45000 nM T96144 C2V5ER 15224740 EC50 = 1700 nM T96144 CO9Z8U 15224741 EC50 = 12000 nM T96144 C6RY8Q 15224742 EC50 = 20000 nM T96144 C14IJQ 15226989 EC50 = 3900 nM T96144 CJ2I9A 15226990 EC50 = 12000 nM T96144 CMG6U9 15226992 EC50 = 7700 nM T96144 CVK0J7 15226993 EC50 = 14000 nM T96144 CQ9D4O 15226994 EC50 = 14000 nM T96144 CM7L0E 15226995 EC50 = 14000 nM T96144 C8BC2I 16092339 IC50 = 226 nM T96144 C3D7WE 17874201 EC50 > 50000 nM T96144 CI0E2S 18654132 EC50 = 500 nM T96144 CM9KB5 19013347 EC50 = 1200 nM T96144 C3AZJ2 19037238 EC50 > 50000 nM T96144 CW0YS3 19977169 IC50 = 3000 nM T96144 C3EHM4 21197160 EC50 > 50000 nM T96144 C3HF6J 23651701 IC50 = 31 ug.mL-1 T96144 COA06G 23692500 EC50 = 74000 nM T96144 C4NB8V 44264761 EC50 = 200000 nM T96144 C1AZ0W 44264768 EC50 = 9100 nM T96144 CZK2G4 44264807 EC50 > 230000 nM T96144 C1EJM2 44264825 EC50 > 210000 nM T96144 CMI89R 44264828 EC50 = 4700 nM T96144 CMDF02 44264839 EC50 = 5100 nM T96144 C0GI4M 44264845 EC50 = 5100 nM T96144 CF0Z5Q 44264850 EC50 > 100000 nM T96144 CDN40P 44264851 EC50 = 2100 nM T96144 CXZS24 44264862 EC50 = 7200 nM T96144 C03DRS 44264866 EC50 > 210000 nM T96144 CV9D7H 44264867 EC50 = 360 nM T96144 CI59CX 44264872 EC50 = 3300 nM T96144 CH6D8L 44264877 EC50 = 6800 nM T96144 CGWJ57 44264878 EC50 = 330 nM T96144 C7TKO2 44264881 EC50 = 98 nM T96144 C60HDJ 44264883 EC50 > 120000 nM T96144 CYNA92 44264901 EC50 = 1600 nM T96144 CW3H1I 44264902 EC50 = 1100 nM T96144 CS3A8Z 44264910 EC50 = 1100 nM T96144 C78NYJ 44264915 EC50 = 160 nM T96144 CL74DG 44264916 EC50 = 160 nM T96144 CF47BK 44264968 EC50 > 120000 nM T96144 C8PT0I 44273491 EC50 > 50000 nM T96144 CS6NT3 44273526 EC50 > 50000 nM T96144 CG8H3R 44273527 EC50 > 50000 nM T96144 C1WAE7 44273560 EC50 > 50000 nM T96144 CQEW06 44273561 EC50 > 50000 nM T96144 CUG08T 44273597 EC50 > 50000 nM T96144 CIC13W 44273598 EC50 > 50000 nM T96144 CC8W2J 44273599 EC50 > 50000 nM T96144 CR1M9A 44273600 EC50 > 50000 nM T96144 CE6F2M 44273605 EC50 > 50000 nM T96144 CBV2Y3 44273617 EC50 > 50000 nM T96144 CAK08Y 44273618 EC50 > 50000 nM T96144 CZ6SM5 44273624 EC50 > 50000 nM T96144 CA8J9D 44273646 EC50 > 50000 nM T96144 CI72SY 44273652 EC50 > 50000 nM T96144 CA6LH1 44273654 EC50 > 50000 nM T96144 C8U2RI 44273699 EC50 > 50000 nM T96144 CY9LQ3 44273700 EC50 > 50000 nM T96144 C09JPK 44290621 IC50 = 220 nM T96144 C28NJR 44292144 EC50 = 62000 nM T96144 CL37PN 44292318 EC50 = 150000 nM T96144 CHT6S2 44292319 EC50 = 510000 nM T96144 CEG4N0 44292374 EC50 = 730000 nM T96144 C3DG7E 44292541 EC50 > 290000 nM T96144 CZB29S 44292578 EC50 = 58000 nM T96144 CT7L9H 44292646 EC50 = 57000 nM T96144 C7IF9P 44292667 EC50 > 130000 nM T96144 CMR8K2 44316531 IC50 = 63 ug.mL-1 T96144 CN9O2M 44328704 IC50 > 400 ug.mL-1 T96144 C7H1SR 44329158 IC50 > 400 ug.mL-1 T96144 CV7PD2 44338996 IC50 = 50000 nM T96144 CK1AF2 44339222 IC50 > 100000 nM T96144 C03KCL 44339290 IC50 = 20000 nM T96144 CEQ3K9 44339418 IC50 > 100000 nM T96144 CJZ07M 44339644 IC50 > 100000 nM T96144 C3C6KN 44339652 IC50 = 50000 nM T96144 CCP1Q4 44342018 IC50 = 17300 nM T96144 CVEO95 44342104 IC50 = 15100 nM T96144 CHAX60 44352794 EC50 = 76000 nM T96144 CTY3D4 44352808 EC50 = 4800 nM T96144 CIUP01 44352809 EC50 = 6300 nM T96144 CG0D1S 44352822 EC50 = 3200 nM T96144 CE5NK3 44352823 EC50 = 5500 nM T96144 C16FRU 44352824 EC50 = 3100 nM T96144 CRL8Q5 44352825 EC50 = 16000 nM T96144 CJ45ZR 44352833 EC50 = 1900 nM T96144 C3HBI2 44352834 EC50 = 92000 nM T96144 CQ1XJ3 44352840 EC50 = 3600 nM T96144 CWT93R 44352841 EC50 = 14000 nM T96144 CC9G2Q 44352850 EC50 = 2600 nM T96144 C2KY4Q 44352857 EC50 = 2400 nM T96144 CSBC36 44352907 EC50 = 7600 nM T96144 C2GZ7E 44352936 EC50 = 2700 nM T96144 C5G0ZS 44352952 EC50 = 4000 nM T96144 CH9UF6 44352953 EC50 = 2300 nM T96144 CX9Y1J 44353051 EC50 = 3800 nM T96144 CC15RG 44353054 EC50 = 9400 nM T96144 CL97SM 44353499 EC50 = 900 nM T96144 CVWY40 44353548 EC50 = 7400 nM T96144 CWDO54 44353588 EC50 = 3200 nM T96144 CA20OD 44353638 EC50 = 6100 nM T96144 C0HXQ4 44353647 EC50 = 1700 nM T96144 CH78SF 44353648 EC50 = 3100 nM T96144 C8QPD4 44353654 EC50 = 1700 nM T96144 CUYJ90 44353655 EC50 = 6400 nM T96144 CPEW14 44353667 EC50 = 3300 nM T96144 C0Q1CK 44353715 EC50 = 11000 nM T96144 CXQ5D4 44353853 EC50 = 5900 nM T96144 CC90EW 44353863 EC50 = 10000 nM T96144 CTR1H5 44355186 EC50 > 50000 nM T96144 C1S7UQ 44355276 EC50 > 50000 nM T96144 CM8QH9 44355294 EC50 > 50000 nM T96144 C0JNW8 44355295 EC50 > 50000 nM T96144 CGFJ50 44355298 EC50 > 50000 nM T96144 C2T8XD 44355299 EC50 > 50000 nM T96144 CC6A2E 44355300 EC50 > 50000 nM T96144 CO2PA6 44355373 EC50 > 50000 nM T96144 C01IZY 44355546 EC50 > 50000 nM T96144 C1CF8Z 44355547 EC50 > 50000 nM T96144 CJ47TM 44356604 IC50 = 720 nM T96144 C8GWD3 44356605 IC50 = 440 nM T96144 C72YUH 44356807 IC50 = 1220 nM T96144 C9J4TH 44356834 IC50 = 420 nM T96144 CNBK67 44358947 EC50 > 100000 nM T96144 CE84TD 44359032 EC50 > 100000 nM T96144 CJ69EP 44359074 EC50 > 100000 nM T96144 CLD4N5 44359075 EC50 = 56000 nM T96144 CXUH17 44359112 EC50 > 100000 nM T96144 CP2L7G 44359116 EC50 > 100000 nM T96144 C4XL7W 44359157 EC50 = 5600 nM T96144 CUI05T 44359158 EC50 > 1000 nM T96144 CCSZ20 44359159 EC50 > 1000 nM T96144 CF7YI0 44387020 EC50 = 21000 nM T96144 C4X2AK 44394836 IC50 = 7 ug.mL-1 T96144 CJRG15 44394923 IC50 = 50.22 ug.mL-1 T96144 C38NBJ 44394954 IC50 = 4.66 ug.mL-1 T96144 CD43AG 44394975 IC50 = 22.47 ug.mL-1 T96144 CP1F2S 44394985 IC50 = 21.89 ug.mL-1 T96144 CIP25C 44395010 IC50 = 6.65 ug.mL-1 T96144 CG9S8U 44396484 IC50 > 500000 nM T96144 CSQ5K2 44396511 IC50 > 500000 nM T96144 CC2AE1 44396529 IC50 > 500000 nM T96144 C0GDR1 44396563 IC50 > 500000 nM T96144 CK8ZW1 44396581 IC50 > 500000 nM T96144 CE04QD 44396595 IC50 > 500000 nM T96144 CEA84D 44399306 IC50 = 66510 nM T96144 C9PYG5 44399370 IC50 = 149970 nM T96144 CI6M1H 44399372 IC50 = 22700 nM T96144 C9P7BU 44399396 IC50 = 23800 nM T96144 CES8H5 44399445 IC50 = 18270 nM T96144 CD4EA8 44399503 IC50 = 83230 nM T96144 CYI0E8 44399554 IC50 = 106800 nM T96144 CP5O2V 44399556 IC50 = 1860 nM T96144 C3DOT7 45260072 EC50 > 560000 nM T96144 C0I1AF 45261142 EC50 > 140000 nM T96144 C8IE5P 45263084 IC50 = 3000 nM T96144 CK7HM1 49796854 IC50 = 1500 nM T96144 C8JQH2 49796857 IC50 = 20000 nM T96144 CT3U6N 49796859 IC50 = 25000 nM T96144 CDS0C6 66825540 IC50 > 500000 nM T96144 C5H6YW 70683609 EC50 > 50000 nM T96144 C9DY6C 76318645 IC50 = 62000 nM T96144 CQ29OX 76325888 IC50 > 500000 nM T96144 CG5QO2 135449100 IC50 = 25000 nM T96144 C68TFR 135457794 IC50 = 25000 nM T96144 CX6F2R 135462833 IC50 > 400 ug.mL-1 T96144 CAEZ52 135972431 IC50 = 25000 nM T96144 CHUO65 136056123 EC50 = 1400 nM T96144 CD1G2J 136056124 EC50 = 1600 nM T96144 C0INA4 136092232 IC50 = 5000 nM T96144 C8RWK6 141750621 IC50 = 23600 nM T96144 C1QP7O 141750622 IC50 = 13700 nM T96144 C3T9YI 141750623 IC50 > 50000 nM T96144 CC56VN 141750625 IC50 = 34800 nM T96144 CT79AN 141750627 IC50 = 12500 nM T96144 C9GX2C 141750629 IC50 > 50000 nM T96144 C4D6SO 141750630 IC50 = 13700 nM T96144 C4I2VY 141750632 IC50 = 16600 nM T96144 CR89LA 141750633 IC50 = 25100 nM T96144 C3I1FN 141750634 IC50 = 17750 nM T96144 CD0BZ2 141750635 IC50 = 13700 nM T96144 CZ8IX7 141750636 IC50 = 23900 nM T96144 C8AXR4 141750637 IC50 = 16100 nM T96144 CT58MU 155514041 IC50 = 116500 nM T96144 COG31S 155514999 IC50 = 12800 nM T96144 CJBE61 155524820 IC50 = 4950 nM T96144 CO3GX9 155532501 IC50 = 124200 nM T96144 CNGX84 155533637 IC50 = 230 nM T96144 C4TRF0 155534357 IC50 = 440 nM T96144 CAC74K 155535167 IC50 = 15400 nM T96144 CVJ20A 155552253 IC50 = 12600 nM T96144 C3XRU8 155560682 IC50 > 50000 nM T96144 CCWE20 155566929 IC50 > 50000 nM T96144 D00DXV 9895647 IC50 = 60 ug.mL-1 T96144 D02DLW 5997 IC50 > 500000 nM T96144 D0NW9G 380482 IC50 = 1000 nM T96144 D0Y6OK 6688 IC50 > 200000 nM T46040 D0I0RJ 16231 IC50 > 50000 nM T46040 D01MUU 183797 IC50 = 20000 nM T46040 D05TKW 16098914 IC50 = 30 nM T46040 CS12YK 80289 IC50 = 120000 nM T46040 CZP0Y1 204101 Ki > 12000 nM T46040 CW93JB 326646 Ki = 70000 nM T46040 C2KYC7 2734311 IC50 = 77300 nM T46040 C7SYK9 6102731 IC50 = 3900 nM T46040 CSQ54Z 6857700 IC50 = 250 nM T46040 C7I5RG 9892392 Ki > 19000 nM T46040 CX85LD 9954980 Ki > 15000 nM T46040 C8L7HY 10097631 Ki = 0.39 nM T46040 CFIH78 10185526 IC50 = 4600 nM T46040 CQ9ZO1 10275412 Ki > 15000 nM T46040 CES6C2 10345244 Ki = 3900 nM T46040 CVK4L6 10418061 IC50 = 24000 nM T46040 CEI65Z 10483775 Ki = 0.2 nM T46040 CLA93S 11237163 Ki > 15000 nM T46040 CRDU42 11271947 Ki > 33000 nM T46040 C73WSC 11273795 IC50 = 63 nM T46040 C68PRG 11341176 IC50 = 116 nM T46040 CR8NW9 11351302 Ki > 10000 nM T46040 CR9Q3O 11399867 IC50 = 12 nM T46040 C6MPD8 11408882 IC50 = 425 nM T46040 C9BO1R 11496443 Ki = 13 nM T46040 CK34OX 11509611 Ki = 120 nM T46040 CTKP68 11518738 Ki = 12 nM T46040 CO68MA 11524737 Ki = 230 nM T46040 C49NVP 11525664 Ki = 9.2 nM T46040 C69FBI 11532883 Ki = 7.5 nM T46040 C3COU7 11553730 Ki = 113 nM T46040 C1VF0M 11561600 Ki = 3.2 nM T46040 CKS10Z 11568460 Ki = 479 nM T46040 CLD19K 11575536 Ki = 56 nM T46040 COW27H 11576157 Ki = 205 nM T46040 C8O1KS 11604020 Ki = 377 nM T46040 C8G7JN 11619799 Ki = 5.3 nM T46040 CXU1Y5 11640546 Ki = 24 nM T46040 C7GUX8 11647632 Ki = 1690 nM T46040 C20JZS 11648035 Ki = 206 nM T46040 CMP2I3 11655755 Ki = 97 nM T46040 C3YAZ2 11668754 Ki = 936 nM T46040 CQHP17 11669959 Ki = 53 nM T46040 CU02GY 11683709 Ki = 949 nM T46040 CJP9O1 11684611 Ki = 0.31 nM T46040 CFDP02 11697636 Ki = 227 nM T46040 CXHC25 11698163 Ki = 61 nM T46040 C9QZY7 11720429 Ki = 58 nM T46040 C69HNO 11984565 Ki = 11000 nM T46040 CT7IR8 12110710 IC50 = 12000 nM T46040 CA86KZ 15947513 Ki = 11000 nM T46040 CU0O5N 15947601 Ki = 11000 nM T46040 CQ3RF8 15947602 Ki = 9700 nM T46040 CS8HY6 15947811 Ki = 11000 nM T46040 CCMQ45 15947923 Ki = 11000 nM T46040 CUGI75 15947926 Ki = 7900 nM T46040 CSV70B 15948627 Ki = 4000 nM T46040 CDSM46 16098887 IC50 = 93 nM T46040 CFK98M 16098895 IC50 = 200 nM T46040 C6BQ0G 16098896 IC50 = 340 nM T46040 C1ZXL4 16098897 IC50 = 710 nM T46040 CP6Y7Q 16098898 IC50 = 920 nM T46040 C3J6LO 16098899 IC50 = 9200 nM T46040 CQ4YJ8 16098900 IC50 = 10 nM T46040 CDL2X5 16098901 IC50 = 45 nM T46040 C53ZXO 16098902 IC50 = 114 nM T46040 CUJ5A9 16098903 IC50 = 136 nM T46040 C0ZWI3 16098904 IC50 = 356 nM T46040 CZ3WM4 16098905 IC50 = 26000 nM T46040 CVN8Y1 16098906 IC50 = 10 nM T46040 CTY5W9 16098907 IC50 = 132 nM T46040 CSBT08 16098908 IC50 = 28 nM T46040 CR9DT0 16098909 IC50 = 533 nM T46040 C53YRO 16098910 IC50 = 6 nM T46040 C91CQM 16098911 IC50 = 7 nM T46040 C0W5NR 16098912 IC50 = 8 nM T46040 CS21OE 16098913 IC50 = 29 nM T46040 CWA54F 16127742 Ki = 330 nM T46040 CDYF29 23646329 IC50 = 76 nM T46040 CKH4O5 24180463 Ki = 7380 nM T46040 C6F8UV 24738839 Ki = 1063 nM T46040 C72BPJ 24738840 Ki = 2530 nM T46040 C5X3YS 24765517 Ki = 3.4 nM T46040 CB29NX 24765713 Ki = 1.9 nM T46040 CJSO87 24849206 Ki > 33000 nM T46040 COX4A7 24873356 Ki = 9100 nM T46040 C9SZ0V 24881874 IC50 = 27000 nM T46040 C19TQN 24881875 IC50 = 1300 nM T46040 CN0ZW3 24999867 Ki > 1000 nM T46040 CEM32W 25001205 Ki > 1000 nM T46040 C4Q9XM 25166807 Ki = 17.5 nM T46040 CX6A4M 25166808 Ki = 47 nM T46040 C2H4PJ 25166809 Ki = 2 nM T46040 CF1I6Q 25166810 Ki = 45.6 nM T46040 C9W0GO 25167018 Ki = 40.5 nM T46040 CE67KP 25252725 Ki = 42 nM T46040 C1SNW5 25253019 Ki = 21 nM T46040 CLWP32 25253020 Ki = 6160 nM T46040 C5W1DZ 44330605 IC50 > 133000 nM T46040 C6B0DP 44330620 IC50 > 133000 nM T46040 C6SV1C 44387258 IC50 = 3900 nM T46040 C0P5DF 44411549 IC50 = 12500 nM T46040 C6M9KP 44411550 IC50 = 2320 nM T46040 C9F4LI 44411551 IC50 = 6220 nM T46040 CX2ZN0 44411553 IC50 = 1200 nM T46040 C7UYQ3 44411556 IC50 = 123000 nM T46040 C4TLD2 44411560 IC50 > 200000 nM T46040 CSG92P 44411585 IC50 = 713 nM T46040 CFCU19 44411590 IC50 = 3310 nM T46040 CP95IE 44411636 IC50 = 431 nM T46040 C40HSW 44411666 IC50 = 1750 nM T46040 C1F2JK 44411677 IC50 = 86000 nM T46040 C68AZJ 44411687 IC50 = 5900 nM T46040 C4GK7S 44411777 IC50 = 790 nM T46040 C0A5GX 44411779 IC50 = 37900 nM T46040 CB34IQ 44411800 IC50 = 2250 nM T46040 C59JRY 44411808 IC50 = 250000 nM T46040 CJU9N6 44411817 IC50 = 1720 nM T46040 C4W5RB 44411818 IC50 = 956 nM T46040 CAT58J 44411821 IC50 > 250000 nM T46040 C3BX5Y 44412781 Ki > 150000 nM T46040 CJ20PN 44416510 IC50 = 24700 nM T46040 CZK3N4 44416547 IC50 = 7300 nM T46040 CQA4B5 44416549 IC50 = 5900 nM T46040 CMVF02 44416571 IC50 = 1400 nM T46040 C3TJK6 44418750 IC50 = 93 nM T46040 C7LK8E 44418751 IC50 = 160 nM T46040 C9G1VL 44418752 IC50 = 258 nM T46040 CHK10G 44418753 IC50 = 403 nM T46040 C9OZ1M 44418754 IC50 = 1920 nM T46040 CE6F4C 44418755 IC50 = 2200 nM T46040 CON3T2 44418756 IC50 = 2600 nM T46040 CE05TM 44418757 IC50 = 2300 nM T46040 CVO5Q1 44432538 Ki > 10000 nM T46040 CQIX73 44434809 Ki > 11000 nM T46040 C5R8HJ 44434815 Ki > 11000 nM T46040 COG34X 44434818 Ki = 10170 nM T46040 C9T1DP 44434835 Ki = 6680 nM T46040 C0L4EK 44453237 IC50 = 10 nM T46040 C59RJK 44453326 IC50 = 850 nM T46040 C8PYF5 44453328 IC50 = 480 nM T46040 C53OJA 44453367 IC50 = 502 nM T46040 CVZW52 44537923 IC50 = 4600 nM T46040 C7K6JN 44587263 Ki = 113 nM T46040 CKL1J2 44587264 Ki = 33 nM T46040 CTF79D 44587290 Ki = 17 nM T46040 CBXY02 44587291 Ki = 259 nM T46040 CDBV80 44587292 Ki = 323 nM T46040 CWZ34J 44587314 Ki = 115 nM T46040 CEXO72 45261244 IC50 = 35000 nM T46040 CNVR31 46905372 IC50 > 133000 nM T46040 CLOY62 49864459 Ki > 33000 nM T46040 CR8JK9 49864483 Ki > 33000 nM T46040 CVD91F 50908869 IC50 = 103100 nM T46040 C1FL6J 52941173 IC50 = 767800 nM T46040 CV8I3U 52942903 IC50 = 145900 nM T46040 C7HVK0 52943592 IC50 = 175900 nM T46040 C1LEN7 52948297 IC50 = 135800 nM T46040 CA6GQ5 53341037 Ki = 1 nM T46040 CIKQ81 53345652 Ki > 130 nM T46040 C7YUN4 53358697 Ki = 636 nM T46040 COT1V5 53358823 Ki = 87 nM T46040 C4QZ2G 53358825 Ki = 42 nM T46040 C96LJG 53358827 Ki = 420 nM T46040 C9BK0S 53358946 Ki = 250 nM T46040 CKY2V1 53392252 IC50 = 9700 nM T46040 CV60BK 53488415 Ki = 13330 nM T46040 CI2ND0 54741583 Ki = 11.2 nM T46040 CU9S6K 57842710 Ki = 10800 nM T46040 CL8T7M 57842742 Ki = 5700 nM T46040 CB5F0H 57942680 Ki = 11000 nM T46040 C8GXF1 57942687 Ki = 11000 nM T46040 CO52PA 57942693 Ki = 11000 nM T46040 CS23DW 57942743 Ki = 11000 nM T46040 C0DO5P 57942817 Ki = 7100 nM T46040 CV0KZ6 57942834 Ki = 2700 nM T46040 C0KRC1 57942835 Ki = 11000 nM T46040 CN7J2K 57976227 Ki = 0.7 nM T46040 CC45OY 57976282 Ki = 0.3 nM T46040 CMDH58 57976350 Ki = 2.4 nM T46040 C9HA0P 57976362 Ki = 422 nM T46040 C60HCV 57976401 Ki = 2.7 nM T46040 CHB27Y 57976410 Ki = 23 nM T46040 CTQ0H4 57976412 Ki = 0.4 nM T46040 CM8UJ7 57976444 Ki = 1.2 nM T46040 CQ71KE 57976446 Ki = 6.7 nM T46040 C3OA5C 58789089 Ki = 6700 nM T46040 C2W1UT 58789135 Ki = 11000 nM T46040 CT9C1Z 58789193 Ki = 11000 nM T46040 CSC0L5 59020200 Ki > 15000 nM T46040 C91APY 59095797 IC50 = 10900 nM T46040 C69SED 59095888 IC50 = 7200 nM T46040 CI4RA5 59158230 Ki = 0.6 nM T46040 CL42XV 59401924 Ki = 173 nM T46040 CHJI56 59401943 Ki = 6.4 nM T46040 CA76HG 59401978 Ki = 3.4 nM T46040 CO38AC 59402011 Ki = 1.6 nM T46040 CVG75I 59402039 Ki = 1.4 nM T46040 CF26ZO 59402046 Ki = 1656 nM T46040 C7IWJ3 59402077 Ki = 5.8 nM T46040 CTW85S 59402125 Ki = 43 nM T46040 CKX9B7 59402220 Ki = 1.7 nM T46040 CZD0N4 59402226 Ki = 2688 nM T46040 CK7I1A 59402239 Ki = 17 nM T46040 C6JP8Q 60154989 Ki = 0.2 nM T46040 CE5A7B 60162406 Ki = 4700 nM T46040 CWCA65 66573845 IC50 > 500000 nM T46040 C3LT2W 66674079 Ki = 590 nM T46040 CYH7X1 66674212 Ki = 1440 nM T46040 C3ND0L 66674351 Ki = 980 nM T46040 C5N1GU 66674475 Ki = 1640 nM T46040 C23QOJ 66674821 Ki = 800 nM T46040 C6AN4O 66698546 Ki = 11 nM T46040 CQM82G 66743646 Ki = 0.69 nM T46040 C3OXF6 66743824 Ki = 0.03 nM T46040 CGS65Y 66743898 Ki = 514 nM T46040 CF41SE 66744041 Ki = 159 nM T46040 CP51WF 66744064 Ki = 5.9 nM T46040 CVJN72 66744470 Ki = 184 nM T46040 CUVZ02 66744488 Ki = 0.88 nM T46040 C07RYU 66744522 Ki = 600 nM T46040 CS0KR9 66744599 Ki = 3.2 nM T46040 CWOD93 66744646 Ki = 0.16 nM T46040 C5OZA3 66744670 Ki = 1.2 nM T46040 CL50WH 66744738 Ki = 16 nM T46040 C16KQV 66744745 Ki = 3.8 nM T46040 CUV7L6 66744747 Ki = 5.2 nM T46040 CK2HY3 66744810 Ki = 68 nM T46040 CO3Q1S 66744936 Ki = 0.47 nM T46040 CLD28I 66744945 Ki = 3920 nM T46040 CYR6V4 66744978 Ki = 76 nM T46040 CH6VF5 66745200 Ki = 21 nM T46040 C72LDB 66939035 Ki = 19 nM T46040 C1Y6JR 67278603 Ki = 433 nM T46040 CR2FQ3 67279044 Ki = 331 nM T46040 CD2FO6 67364478 Ki = 11423 nM T46040 C3DC0X 68096989 Ki = 264 nM T46040 C4JGQ5 68096996 Ki = 560 nM T46040 CYR28O 68265957 Ki = 92 nM T46040 C84VRW 68265970 Ki = 8.2 nM T46040 C0DXP4 68266030 Ki = 17 nM T46040 C6AM5R 68266034 Ki = 500 nM T46040 CE79VS 68440006 Ki = 11000 nM T46040 CA49UK 69520512 Ki > 19000 nM T46040 CV7O4T 69913810 Ki = 1000 nM T46040 C6X1HO 70252779 Ki = 31 nM T46040 C6AU1R 70252985 Ki = 7 nM T46040 C4LQD6 70253152 Ki = 36 nM T46040 CTO5I6 70253788 Ki = 10 nM T46040 C8A7ZJ 70306716 Ki = 18 nM T46040 C2NWX6 71260289 Ki = 4.8 nM T46040 CUQ69P 71260381 Ki = 99 nM T46040 C9EL3C 71260387 Ki = 17 nM T46040 C1JYH2 71260430 Ki = 0.95 nM T46040 CFLW10 71260451 Ki = 4.7 nM T46040 CBZS27 71260458 Ki = 333 nM T46040 CDXF69 71263009 Ki = 34 nM T46040 C2WX4Y 71263010 Ki = 231 nM T46040 CL5TU2 71263047 Ki = 2890 nM T46040 CQE0M7 71509195 Ki = 5.5 nM T46040 CZ43AI 71509198 Ki = 11 nM T46040 C9E3FW 71509332 Ki = 47 nM T46040 C0CM2A 71509334 Ki = 1390 nM T46040 CWKL95 71543361 Ki = 3.7 nM T46040 C06NDL 71548081 Ki < 5 nM T46040 CJPF90 71548883 Ki = 0.71 nM T46040 CG4UN0 71550253 Ki = 1700 nM T46040 CO1LP3 71550396 Ki = 11 nM T46040 C9FRP5 71550399 Ki = 290 nM T46040 CIY1U2 71550400 Ki = 110 nM T46040 CS5V2J 71550537 Ki = 57 nM T46040 C30ZKJ 71561420 Ki = 3370 nM T46040 C83ZNH 71562308 IC50 = 92.7 ug.mL-1 T46040 C1E3TA 71600123 IC50 > 1000000 nM T46040 C4NTV2 71600125 IC50 = 216000 nM T46040 CPU48B 71600127 IC50 = 407000 nM T46040 CTJ02W 71600261 IC50 = 305000 nM T46040 C9LHZ2 71600263 IC50 = 90000 nM T46040 C0VP6U 71600678 IC50 > 1000000 nM T46040 C5X9VU 71600679 IC50 = 102000 nM T46040 C02PZE 71600941 IC50 = 139000 nM T46040 C64SPE 71600942 IC50 = 320000 nM T46040 C0JB9U 71600943 IC50 = 159000 nM T46040 CU6VX7 71601065 IC50 = 82000 nM T46040 CGV2Y5 71601066 IC50 = 91000 nM T46040 C42VZK 71601067 IC50 = 59000 nM T46040 CDI64Z 71601210 IC50 = 52000 nM T46040 COI0H7 71601211 IC50 = 182000 nM T46040 C90RAW 71601212 IC50 = 213000 nM T46040 CUP95T 71601350 IC50 = 273000 nM T46040 C45PTU 71601351 IC50 > 1000000 nM T46040 CRD4I9 71625797 Ki > 55000 nM T46040 C62ZTJ 71660643 IC50 > 33000 nM T46040 C78DJQ 71711730 IC50 < 10000 nM T46040 CD53RA 71716975 Ki > 120000 nM T46040 CSP5T2 71716976 Ki > 120000 nM T46040 CKY5O6 71718753 IC50 = 153000 nM T46040 CR6S5X 71734401 IC50 = 384000 nM T46040 C0AK9E 71734402 IC50 = 29900 nM T46040 C2XUG1 71734404 IC50 = 29900 nM T46040 C6F8PU 71734497 IC50 = 99000 nM T46040 C08BOY 71734677 IC50 = 6400 nM T46040 CTS91W 71734679 IC50 = 14900 nM T46040 C26QMO 71734771 IC50 = 820 nM T46040 CFJ1W4 71734773 IC50 = 47200 nM T46040 CRBH34 72164200 IC50 > 33000 nM T46040 CWNZ45 72164201 IC50 = 20800 nM T46040 CK34ZH 72550138 Ki > 10000 nM T46040 CT45ER 72550807 Ki = 2900 nM T46040 C46TNC 72550811 Ki = 6100 nM T46040 CLI36U 72551247 Ki = 3400 nM T46040 CAZ5R4 72725806 Ki = 1.5 nM T46040 CPW7T3 72725807 Ki = 7.6 nM T46040 C01LOR 73051877 Ki = 0.08 nM T46040 C6M9ZP 73052197 Ki = 43.82 nM T46040 CXJ86Q 73052510 Ki = 0.11 nM T46040 CB14LR 73052831 Ki = 0.98 nM T46040 CH3A6Q 73332164 Ki = 2.4 nM T46040 CH1BJ2 76311085 Ki = 8.5 nM T46040 C8RYU0 76311086 Ki = 2400 nM T46040 C9OKI1 76311087 Ki = 15 nM T46040 CZU72O 76311088 Ki = 64 nM T46040 CE3ZI8 76311089 Ki = 110 nM T46040 C29QNE 76311090 Ki = 154 nM T46040 C3R8LG 76311091 Ki = 0.64 nM T46040 CUZM48 76314299 Ki > 19000 nM T46040 CRXU73 76314700 Ki = 1960 nM T46040 CSBD17 76314701 Ki = 110 nM T46040 C9J0BH 76317785 Ki = 10000 nM T46040 C9C4BV 76317871 Ki = 19000 nM T46040 CSY3T8 76318271 Ki = 110 nM T46040 CI7MO1 76318272 Ki = 37 nM T46040 C28QGR 76318273 Ki = 540 nM T46040 C4WUP1 76318274 Ki = 26 nM T46040 C9PJ1H 76321975 Ki = 48 nM T46040 C7UP8I 76321976 Ki = 0.3 nM T46040 CO28RN 76325189 Ki = 800 nM T46040 CHNJ05 76325595 Ki = 25 nM T46040 C6UR1G 76325596 Ki = 23 nM T46040 CO3H5T 76328753 Ki > 19000 nM T46040 C3W5PN 76329159 Ki = 61 nM T46040 CJ9D8H 76329160 Ki = 0.72 nM T46040 C6CW8M 76332426 Ki > 19000 nM T46040 CL09IJ 76332819 Ki = 3.9 nM T46040 CXKG18 76332820 Ki = 466 nM T46040 CYCA26 76332821 Ki = 0.69 nM T46040 C0A9XJ 76336440 Ki = 830 nM T46040 CADC95 76336441 Ki = 79 nM T46040 CZ4N5I 76336442 Ki = 207 nM T46040 C7TNX2 76336443 Ki = 1 nM T46040 CAT95V 76685067 IC50 > 100000 nM T46040 CMD5V7 86583041 Ki = 7.2 nM T46040 CF83UD 87114200 Ki = 26 nM T46040 CUS40A 88235291 Ki = 12 nM T46040 CO6U9I 88582319 Ki = 9.6 nM T46040 CVD6W9 88583174 Ki = 10 nM T46040 CPI21N 88983246 Ki = 9.3 nM T46040 CY86FT 89273814 Ki = 1.5 nM T46040 CXBA59 89273816 Ki = 0.53 nM T46040 C7O5LA 89273817 Ki = 0.32 nM T46040 C01JOE 89273818 Ki = 6400 nM T46040 C59WJV 89273819 Ki = 8100 nM T46040 C3JM4Z 89273820 Ki = 71 nM T46040 CZKM65 89501080 Ki = 83 nM T46040 C58RDS 89501761 Ki = 160 nM T46040 C7DEI2 89501771 Ki = 300 nM T46040 CH21ZI 89501772 Ki = 2000 nM T46040 CFQ90S 89501773 Ki = 270 nM T46040 C7YAG4 89501774 Ki = 640 nM T46040 C0MV8C 89501782 Ki = 27 nM T46040 C1J5UP 89501791 Ki = 6 nM T46040 CCAF03 89501798 Ki = 17 nM T46040 CBQM32 89501809 Ki = 80 nM T46040 C70PEJ 89501825 Ki = 51 nM T46040 CV4XK5 89509984 Ki = 5.8 nM T46040 C4BX1G 89510211 Ki = 890 nM T46040 C8OP0Z 89510222 Ki = 1400 nM T46040 C25NOF 89510265 Ki = 870 nM T46040 CAL4P7 89510370 Ki = 39 nM T46040 C5ZO9S 89510407 Ki = 74 nM T46040 CTZ95F 90411167 Ki = 23 nM T46040 CMFV97 90411307 Ki = 21 nM T46040 C9P5VD 90454231 Ki = 29 nM T46040 CER1Y7 90478342 Ki = 5 nM T46040 CQG9T0 90480064 IC50 = 2800 nM T46040 CM5S1Z 90655980 IC50 = 7500 nM T46040 CZ1NV3 90655982 IC50 = 109000 nM T46040 CGM04C 90655984 IC50 = 122000 nM T46040 COH41Y 91666660 Ki = 0.02 nM T46040 CK3P6X 91667569 IC50 = 0.8 nM T46040 C65TLW 101862198 Ki > 1000000 nM T46040 CL8WC6 117819668 IC50 = 7700 nM T46040 CNY29S 117819734 IC50 = 650 nM T46040 C2W5BU 117820065 IC50 = 4000 nM T46040 CEI6Y5 117820116 IC50 = 2100 nM T46040 CG6S9U 117820135 IC50 > 100000 nM T46040 CI4ZR0 117820213 IC50 = 5200 nM T46040 C2RXZ3 117820231 IC50 = 600 nM T46040 CI5EW6 117820295 IC50 = 8090 nM T46040 C4HAT8 117820303 IC50 = 4800 nM T46040 CJ10KS 117828732 Ki = 1.1 nM T46040 CTAC25 117828738 Ki = 0.39 nM T46040 C98BXU 117984620 IC50 = 14 nM T46040 CH5Z4P 117985339 IC50 = 3.5 nM T46040 CPAC38 117986252 IC50 = 2.8 nM T46040 C3KB4M 117986600 IC50 = 0.9 nM T46040 CI4KC5 117986603 IC50 = 0.34 nM T46040 C3PS6Y 118098650 Ki = 2300 nM T46040 CKS29X 118713018 IC50 > 100000 nM T46040 CRF62H 118713026 IC50 > 100000 nM T46040 CAS3L5 118713029 IC50 > 100000 nM T46040 C3MVG0 118720988 Ki = 495 nM T46040 C9M2IH 118720990 Ki = 1120 nM T46040 C1E6GW 118720991 Ki = 630 nM T46040 C9BVI5 118720993 Ki = 1340 nM T46040 C1FQZ6 118720994 Ki = 30 nM T46040 C0WZA2 118720996 Ki = 350 nM T46040 CE89KB 118720997 Ki = 2860 nM T46040 CIAL50 118720998 Ki = 150 nM T46040 C4HLM3 118720999 Ki = 400 nM T46040 CLD6I3 118721000 Ki = 1100 nM T46040 C0XG7H 118721001 Ki = 275 nM T46040 CZC53M 118721002 Ki = 545 nM T46040 C8FZ2L 118721003 Ki = 9 nM T46040 C0M4IQ 118721004 Ki = 4 nM T46040 CLRB29 118721005 Ki = 3 nM T46040 C9B1FX 118721007 Ki = 3 nM T46040 CRV5Y1 118721008 Ki = 0.3 nM T46040 CH6AQ9 118721009 Ki = 0.3 nM T46040 CKF56V 118723650 IC50 = 6300 nM T46040 C4U2AW 118723894 IC50 = 124000 nM T46040 CV5JG3 118723904 IC50 = 118000 nM T46040 CP98JL 118723906 IC50 = 220000 nM T46040 C0UO7Q 118723908 IC50 = 86900 nM T46040 CGFK89 118725481 Ki = 30207 nM T46040 C34GCZ 118725482 Ki = 12 nM T46040 CHG7C5 118725483 Ki = 320 nM T46040 CY9E0H 118725484 Ki = 860 nM T46040 CQ4LY6 118725485 Ki = 1067 nM T46040 CLA74U 118727593 Ki = 1.49 nM T46040 C79JAG 118727594 Ki = 2900 nM T46040 C0NKE3 118727595 Ki = 68 nM T46040 CHQ5P7 118987013 Ki = 6.3 nM T46040 C2V6PQ 122550396 IC50 = 21.5 nM T46040 C8NR0Y 122550417 IC50 = 6.5 nM T46040 C3W6DG 122551266 IC50 < 0.13 nM T46040 CEXK15 126843252 Ki = 0.5 nM T46040 C5Y8IS 127025168 Ki = 0.36 nM T46040 CY03UC 127027302 Ki = 7.1 nM T46040 C18GDE 127027303 Ki = 11.5 nM T46040 CK0W2P 127027635 Ki = 2 nM T46040 CWJ0Y6 127027636 Ki = 1.8 nM T46040 C36DML 127029802 Ki = 5.5 nM T46040 CLJ40K 127029803 Ki = 14 nM T46040 C60ASZ 127029813 Ki = 9.1 nM T46040 CIUQ08 127029817 Ki = 11 nM T46040 C9MIG8 127030139 Ki = 6.7 nM T46040 CXI04N 127030140 Ki = 3.197 nM T46040 CGT4N5 127030754 Ki = 87 nM T46040 C78TRJ 127030755 Ki = 3.8 nM T46040 CW5N6I 127030756 Ki = 10 nM T46040 C8WO2P 127031081 Ki = 144 nM T46040 CPC0M8 127031390 Ki = 3.7 nM T46040 C9T3VX 127031975 Ki = 87 nM T46040 C8ZUT5 127031976 Ki = 110 nM T46040 CFCD34 127032571 Ki = 17 nM T46040 CVE9J1 127032572 Ki = 8.4 nM T46040 CU6CK8 127032879 Ki = 7.9 nM T46040 C1BWV2 127035672 Ki = 12100 nM T46040 CVRY56 127036086 Ki = 3970 nM T46040 C9B6LT 127037264 Ki = 6630 nM T46040 C60HLK 127037469 Ki = 2560 nM T46040 C4T9KU 127045502 Ki > 11000 nM T46040 C4RFP7 127045503 Ki > 14200 nM T46040 C2IOG9 127045504 Ki > 14200 nM T46040 CHK80O 127045505 Ki > 14200 nM T46040 CL6W5N 127045506 Ki > 14200 nM T46040 C8NDY0 131800962 Ki = 23 nM T46040 COLE34 132585254 Ki = 0.07 nM T46040 CT2RV6 134130781 IC50 = 106000 nM T46040 CWV3G6 134131077 IC50 = 12700 nM T46040 CS8FV1 134131084 IC50 = 40900 nM T46040 C92RTL 134131303 IC50 = 11700 nM T46040 CL37SG 134131589 IC50 = 3610 nM T46040 CPQ04R 134132204 Ki > 10000 nM T46040 C6DPW7 134141496 Ki = 6500 nM T46040 CIRU10 134145163 Ki = 3100 nM T46040 CHA7X9 134146314 Ki = 7100 nM T46040 CAZ1W4 134147472 Ki = 0.5 nM T46040 CTG65U 134148771 Ki = 8800 nM T46040 C3QEO5 134151811 Ki = 1400 nM T46040 C6HTD5 135393470 IC50 = 31000 nM T46040 C7NA6E 135393474 IC50 > 50000 nM T46040 C4CMO6 136003658 Ki = 2 nM T46040 C1GPL0 136402490 Ki = 3074 nM T46040 CEY3Q1 137348813 Ki = 12 nM T46040 CD60AV 137348814 Ki = 0.18 nM T46040 CQ60BM 137348815 Ki = 0.13 nM T46040 CC3LM9 137631467 Ki = 0.07 nM T46040 C9TF6L 137631761 Ki = 35 nM T46040 C2JT1W 137632528 IC50 = 208000 nM T46040 CL9E3H 137632768 Ki = 44 nM T46040 CV91SN 137633060 Ki = 2200 nM T46040 CX19QM 137634842 Ki = 17 nM T46040 C3B0ZQ 137635582 Ki = 6.5 nM T46040 C2NCF1 137635772 Ki = 0.33 nM T46040 C8TP4B 137636329 Ki = 2 nM T46040 CWC51M 137637127 Ki = 6 nM T46040 CDQ62V 137637214 Ki > 50000 nM T46040 CGBF35 137638492 Ki = 230 nM T46040 C2K8JV 137639385 Ki = 500 nM T46040 CH47NJ 137643037 Ki = 1.4 nM T46040 CO7G6Q 137643614 Ki = 0.49 nM T46040 C4R7GB 137644296 Ki < 5 nM T46040 C2E7DK 137645204 Ki = 18 nM T46040 CCW60X 137646972 Ki = 17 nM T46040 CNO2T8 137647340 IC50 = 180000 nM T46040 C3JO2N 137647396 Ki = 28 nM T46040 CB1F6T 137648063 Ki = 7 nM T46040 CX8W2I 137648336 Ki = 1.4 nM T46040 C3LMV5 137648502 Ki = 12 nM T46040 CGU24V 137648949 Ki = 10 nM T46040 C4ZCU8 137649155 Ki = 0.38 nM T46040 CGWB41 137651065 Ki = 2.2 nM T46040 C38AWX 137651505 Ki = 25 nM T46040 C3QSL4 137651514 Ki = 27 nM T46040 C39OVW 137652569 Ki = 2 nM T46040 CLG07H 137653868 Ki = 27 nM T46040 CNX46H 137654508 Ki > 50000 nM T46040 C3Y1VG 137656151 Ki = 21 nM T46040 CKV94N 137657082 Ki = 0.14 nM T46040 CU6JS9 137657273 Ki = 400 nM T46040 CU34XV 137658570 Ki = 2 nM T46040 CU9NX0 137659435 Ki = 0.098 nM T46040 CFZ53J 137659839 Ki = 25 nM T46040 C2TD1I 137660311 Ki = 140 nM T46040 C1JQX3 137662013 Ki = 0.06 nM T46040 CO51HN 139030452 IC50 > 50000 nM T46040 C10JPH 139208763 Ki = 2.1 nM T46040 CX07YE 139592452 Ki = 5.3 nM T46040 C7XW0S 140560726 Ki = 10 nM T46040 C0XH7T 145967687 Ki = 89 nM T46040 CI87RZ 145968383 Ki = 6.1 nM T46040 C3SI6F 145969531 Ki = 22 nM T46040 C5NE8Z 145970200 Ki = 4.1 nM T46040 CHC18Z 145970336 Ki = 6.6 nM T46040 CE6C0A 145970642 Ki = 1.9 nM T46040 CTOX41 145977265 Ki = 0.3 nM T46040 CZ1R3B 145982984 Ki = 18 nM T46040 CGP50S 145986794 Ki = 4 nM T46040 C4HLX8 146029523 IC50 = 23300 nM T46040 CICU31 155511394 Ki = 1936 nM T46040 C3U8GK 155511607 IC50 = 0.7 nM T46040 CV7QT3 155512262 Ki = 3.4 nM T46040 C2VX3G 155512946 Ki = 4.1 nM T46040 C50SFE 155513574 Ki = 871 nM T46040 C2CI8S 155513907 Ki = 1697 nM T46040 CYT20V 155514020 Ki > 50000 nM T46040 C9ZF3E 155514138 Ki = 0.18 nM T46040 CAT98N 155514640 Ki > 10000 nM T46040 CK8AZ9 155514961 Ki = 189 nM T46040 CPUG37 155516479 Ki > 19000 nM T46040 CV0A7G 155517265 Ki = 0.2 nM T46040 CT5XA7 155517793 Ki = 38 nM T46040 CF96DM 155518671 Ki > 10000 nM T46040 C7DUX3 155520916 Ki > 10000 nM T46040 CGKD97 155523007 Ki = 1.8 nM T46040 CAL0O2 155524490 Ki = 372 nM T46040 CUQZ15 155528151 Ki = 2.2 nM T46040 CEU02X 155530331 Ki > 13300 nM T46040 C46AZL 155530642 Ki > 25000 nM T46040 CX7Z5A 155530964 Ki = 4.4 nM T46040 CATX95 155535014 Ki = 7 nM T46040 C6RW8T 155537983 Ki = 2.1 nM T46040 C7YUJ9 155539325 Ki = 201 nM T46040 CL90DN 155540666 Ki > 10000 nM T46040 C4P2GV 155543617 Ki > 25000 nM T46040 CVJE95 155547007 Ki = 2.2 nM T46040 CU9FL4 155551858 Ki > 50000 nM T46040 CIS87V 155552284 Ki = 175 nM T46040 CUN0O2 155553801 Ki = 0.27 nM T46040 CX2Y0Q 155555090 Ki = 1.8 nM T46040 CU8LR3 155555208 Ki > 25000 nM T46040 C5YE0M 155567050 Ki = 45 nM T46040 CP4F1U 155567613 Ki = 13000 nM T46040 CEZ8B9 155568406 Ki > 100000 nM T46040 CD81GH 46830813 IC50 = 3.9 nM T46040 D02AVL 18376720 Ki > 5000 nM T46040 D02PAU 16731825 Ki > 10000 nM T46040 D02YIW 1794 IC50 > 50000 nM T46040 D09YQM 9802488 IC50 = 2.8 nM T46040 D0ON2Z 204102 Ki > 12000 nM T46040 D0R9CH 3400921 Ki > 10000 nM T46040 D0V7TH 76328755 Ki = 300 nM T46040 D0Y5IQ 44255320 IC50 = 10000 nM T34123 D0C7ET 11174599 IC50 < 30 nM T34123 C7AYV5 118540795 IC50 > 10000 nM T34123 D0P8TL 56947150 IC50 > 10000 nM T88947 D0YV1Q 6032 IC50 = 9400 nM T88947 C2I9SB 145963963 IC50 = 6200 nM T88947 CNO5R6 145964081 IC50 = 13500 nM T88947 C9JQ7U 145964160 IC50 = 8400 nM T88947 C1HG0J 145964452 IC50 = 6600 nM T88947 CA49KD 145965656 IC50 = 8100 nM T88947 CB37JH 145966327 IC50 = 4900 nM T88947 C2D4CT 145967368 IC50 = 6200 nM T88947 C9BIJ1 145972607 IC50 = 13000 nM T88947 C2F8DM 145973926 IC50 = 13600 nM T88947 CYC2H4 145974601 IC50 = 18800 nM T88947 CCP06R 145976504 IC50 = 7600 nM T88947 CC7GN6 145976576 IC50 = 2500 nM T88947 CG71VQ 145977097 IC50 = 4300 nM T88947 CF7OZ3 145977387 IC50 = 19000 nM T00488 CQTJ86 9547099 EC50 = 28 nM T00488 CIY57T 9547100 EC50 = 25.7 nM T00488 C6L2IH 44475675 EC50 = 87 nM T00488 CE2FR8 52926276 EC50 = 933.25 nM T00488 CK6IV9 52926277 EC50 = 72 nM T00488 CSV34F 52926278 EC50 = 85.11 nM T00488 CJI7F3 71495077 EC50 = 25 nM T00488 CX0L7E 101780959 EC50 = 2200 nM T00488 C48ZQW 101780960 EC50 > 1000 nM T00488 CVM0N2 122177490 EC50 = 38.9 nM T00488 C5U2LP 122177491 EC50 > 1000 nM T00488 C02ODQ 122177492 EC50 = 58 nM T00488 C0PF6Z 122177493 EC50 = 144.54 nM T00488 CQ4H8Y 122177494 EC50 > 1000 nM T00488 CY7PH9 122177495 EC50 = 645.65 nM T00488 CW9OA2 122177496 EC50 > 1000 nM T00488 CC43DK 122177497 EC50 = 57.54 nM T00488 C2BWT6 122177498 EC50 = 21 nM T00488 C4C1RL 122177499 EC50 = 44.67 nM T00488 CC7DB0 122177500 EC50 = 520 nM T00488 CH69GX 122177501 EC50 = 400 nM T00488 C51KDV 122177502 EC50 = 169.82 nM T00488 C5L3NY 122177503 EC50 = 4466.84 nM T00488 CEZN81 122177504 EC50 = 1148.15 nM T00488 C0L7DS 122177505 EC50 = 330 nM T00488 C6GHW5 122177506 EC50 = 140 nM T00488 CIR31U 122177507 EC50 > 1000 nM T00488 C9ZO0D 122177508 EC50 > 1000 nM T00488 CAE7Y0 122177509 EC50 = 2041.74 nM T00488 COD16Y 122177510 EC50 = 210 nM T00488 CBI02Q 122177511 EC50 = 707.95 nM T00488 C2TQ8R 122177513 EC50 = 120 nM T00488 CA0T9U 122177514 EC50 = 100 nM T00488 CZY0A1 122177515 EC50 = 457.09 nM T00488 CAZ90F 122177516 EC50 = 3.162 nM T00488 C4JP1B 122177517 EC50 = 1.995 nM T00488 C2GY9U 122177518 EC50 = 12 nM T00488 CX5EK3 122177519 EC50 = 83 nM T00488 CLD62P 122177520 EC50 = 2.63 nM T00488 CA8ZJ5 122177521 EC50 = 12.88 nM T00488 C67LAE 122177522 EC50 = 53 nM T00488 C30HEC 122177523 EC50 = 85.11 nM T00488 CJ0RD5 122177524 EC50 = 3.7 nM T00488 C6GI8E 122177525 EC50 = 1.698 nM T00488 C0C5XU 122177526 EC50 = 32.36 nM T00488 C74WRP 122177527 EC50 = 54.95 nM T00488 C61RUZ 122177528 EC50 = 1.3 nM T00488 CRZ1V8 122177589 EC50 = 3.3 nM T00488 C8XY1C 122177590 EC50 = 549.54 nM T00488 C6SGF5 122177591 EC50 > 1000 nM T00488 CFLM72 122177592 EC50 > 1000 nM T98896 D05VZE 119031 IC50 = 10000 nM T98896 D0G1LL 74221072 IC50 = 2 nM T98896 D0N6ZA 74221131 IC50 = 8 nM T98896 D0UM5R 74221070 IC50 = 4 nM T98896 D0T9HG 132519 IC50 = 500 nM T98896 CR80LA 1268892 IC50 > 22000 nM T98896 CGM37W 1358227 IC50 = 20100 nM T98896 C6UHJ5 1732703 IC50 = 3500 nM T98896 C9CLT4 2897263 IC50 = 760 nM T98896 CR8O7X 2897629 IC50 = 460 nM T98896 CHL07C 2897655 IC50 = 1000 nM T98896 CYH9X4 2897704 IC50 = 830 nM T98896 CT32BN 3136571 IC50 = 9600 nM T98896 C6W4EU 3136575 IC50 = 11100 nM T98896 CY3IC0 3136622 IC50 = 13600 nM T98896 C2NLA8 3136666 IC50 = 3700 nM T98896 CA1XR5 3136667 IC50 = 4600 nM T98896 CU23OK 3136668 IC50 = 1900 nM T98896 CVN4Y1 3137370 IC50 = 12600 nM T98896 C05SVN 3561957 IC50 = 24200 nM T98896 CT8PU3 3671894 IC50 = 350 nM T98896 CV7C5N 3800952 IC50 = 24100 nM T98896 CRAX63 3872724 IC50 = 3000 nM T98896 C35QCG 4606700 IC50 = 780 nM T98896 CY4XN6 5880744 IC50 > 67000 nM T98896 CJS23I 9868333 Ki = 1900 nM T98896 C9X0YR 9954867 IC50 = 12 nM T98896 CN76XI 9957653 IC50 = 420 nM T98896 CV5X8A 10224181 IC50 > 25000 nM T98896 CY08WJ 10322755 Ki = 1900 nM T98896 CG49SC 11201179 IC50 = 84 nM T98896 C8C5AV 11294179 Ki = 1000 nM T98896 C3RJ8Z 11496896 IC50 = 3700 nM T98896 C5MO0U 11526826 IC50 = 2600 nM T98896 CW5A4S 11569716 IC50 = 6600 nM T98896 CRF7V9 11691964 IC50 = 8400 nM T98896 C6HV8Z 11752434 IC50 = 1.4 nM T98896 C6Y7QT 16664963 IC50 = 1100 nM T98896 C0EB1Z 16730403 IC50 = 6700 nM T98896 C4S5KG 19201200 IC50 > 22000 nM T98896 CIC4S9 22004232 IC50 = 3400 nM T98896 C38XLI 22885492 IC50 = 1700 nM T98896 CQE26H 24180584 IC50 = 610 nM T98896 CR5CP6 24677765 IC50 = 5300 nM T98896 CGT06Y 24752936 IC50 = 1400 nM T98896 C5R4BG 24752938 IC50 = 7200 nM T98896 CWH71J 24752939 IC50 = 1200 nM T98896 CGJ0Y5 24753023 IC50 = 1400 nM T98896 CFC84I 24753024 IC50 = 2600 nM T98896 C45NTH 24753026 IC50 = 3100 nM T98896 C21DJN 24753934 IC50 = 7500 nM T98896 CAN0F9 24753935 IC50 = 13400 nM T98896 C2EAY6 24753936 IC50 = 2400 nM T98896 CGQ93N 24753937 IC50 = 2500 nM T98896 C2ANP6 24754101 IC50 = 1500 nM T98896 CU0OI7 24754102 IC50 = 4400 nM T98896 CM8IV9 24754103 IC50 = 2000 nM T98896 CXEP14 24754176 IC50 = 870 nM T98896 CY0D8Z 24754177 IC50 = 1200 nM T98896 CSQ9E4 24754248 IC50 = 780 nM T98896 CG9YV5 24754250 IC50 = 1400 nM T98896 CX16GL 24754251 IC50 = 640 nM T98896 COY8K0 24754252 IC50 = 900 nM T98896 CYW5G8 24901471 IC50 = 950 nM T98896 C7LK3H 24957414 IC50 = 830 nM T98896 CH13AS 24957416 IC50 = 2420 nM T98896 C3VD8K 24957417 IC50 = 1320 nM T98896 C0WAE7 24957794 IC50 = 800 nM T98896 CBC98K 24957795 IC50 = 620 nM T98896 CB3WM1 24957797 IC50 = 990 nM T98896 CF58EN 24957798 IC50 = 1310 nM T98896 C1SZP4 24957799 IC50 = 1890 nM T98896 C90HIA 24958174 IC50 = 1250 nM T98896 CW1E6D 24958175 IC50 = 1440 nM T98896 C1B9WF 24958176 IC50 = 1700 nM T98896 CG78HC 24958177 IC50 = 830 nM T98896 CW5NM7 24958178 IC50 = 780 nM T98896 C4NLR6 24958179 IC50 = 1280 nM T98896 CV0D2I 24958547 IC50 = 1830 nM T98896 CB0OD1 24958548 IC50 = 700 nM T98896 CB94KU 24958549 IC50 = 560 nM T98896 CA82BG 24958550 IC50 = 820 nM T98896 CORS65 24959643 IC50 = 770 nM T98896 CJ0U2Q 24959645 IC50 > 10000 nM T98896 C7KCD4 24959646 IC50 = 1900 nM T98896 CUOD65 24960008 IC50 = 2280 nM T98896 C2ZLB8 24960375 IC50 = 2980 nM T98896 CR52XT 24960376 IC50 = 1670 nM T98896 CU3W7Y 24960377 IC50 = 490 nM T98896 CE0Q8H 24960735 IC50 > 10000 nM T98896 CZ3R4G 24960736 IC50 = 3390 nM T98896 CV5Y6F 24960737 IC50 = 1720 nM T98896 CUX89F 24960738 IC50 > 10000 nM T98896 CSQ1V2 24960739 IC50 > 10000 nM T98896 CZJ97F 24961101 IC50 = 2340 nM T98896 CNA14R 24961102 IC50 = 1850 nM T98896 CA1YC3 24961103 IC50 = 1660 nM T98896 CIMX02 24961104 IC50 = 2330 nM T98896 CI25YZ 24961105 IC50 > 10000 nM T98896 CDEM60 24961464 IC50 > 10000 nM T98896 CVCM56 24961465 IC50 > 10000 nM T98896 C4FWZ0 24961466 IC50 = 1330 nM T98896 C25UWJ 24961468 IC50 = 3370 nM T98896 CE7MA8 24961825 IC50 = 1480 nM T98896 CMR14B 24961829 IC50 = 1010 nM T98896 C0HW6Y 24961830 IC50 = 1120 nM T98896 C9HRX3 24962189 IC50 = 1930 nM T98896 CD0FO1 24962190 IC50 = 1580 nM T98896 C95HGN 24962193 IC50 = 1070 nM T98896 C82YHC 24962547 IC50 = 1190 nM T98896 C7KLT8 24962548 IC50 = 2770 nM T98896 CY5M6H 24962550 IC50 = 1430 nM T98896 CWVZ68 24962551 IC50 = 1220 nM T98896 CC6X1Y 24962552 IC50 = 2320 nM T98896 C5OUQ9 24962913 IC50 = 1210 nM T98896 CVR52U 25066764 IC50 > 10 nM T98896 CHR2P1 25183768 Ki > 25000 nM T98896 CLG95N 25263183 IC50 = 3200 nM T98896 CL6FK4 25263184 IC50 = 8000 nM T98896 CGH9Y7 25263189 IC50 = 7300 nM T98896 CS8X0C 25263190 IC50 = 1600 nM T98896 CMO1F8 25263191 IC50 = 200 nM T98896 CYB7W5 25263193 IC50 = 880 nM T98896 C32HSE 25263196 IC50 = 4500 nM T98896 CXI74K 25263200 IC50 = 310 nM T98896 CZ15TS 25263201 IC50 = 220 nM T98896 C74GMF 25263202 IC50 = 210 nM T98896 CY8V2M 25263203 IC50 = 180 nM T98896 C7YXE1 25263204 IC50 = 78 nM T98896 C0VFD4 25263206 IC50 = 290 nM T98896 CHL68Z 25263211 IC50 = 260 nM T98896 C4DRN5 25263212 IC50 = 270 nM T98896 CLGA45 25263213 IC50 = 270 nM T98896 C0AWF6 27036527 IC50 = 2800 nM T98896 CRD2U0 44201336 IC50 = 71 nM T98896 CCI64J 44224245 IC50 = 22600 nM T98896 CZB81D 44395506 IC50 = 1 nM T98896 C30DKN 44404553 IC50 = 330 nM T98896 C6H9DO 44425389 IC50 = 1800 nM T98896 CM8LF3 44425390 IC50 = 1400 nM T98896 CA26XS 44425391 IC50 = 11600 nM T98896 CU7TS1 44425392 IC50 = 4900 nM T98896 CC0A2L 44425393 IC50 = 16200 nM T98896 CNOK41 44425394 IC50 = 14800 nM T98896 CZ1Y9M 44425395 IC50 = 3200 nM T98896 CQ6TA9 44425396 IC50 = 2500 nM T98896 CKFE92 44425397 IC50 = 5300 nM T98896 CB0SI5 44425398 IC50 > 22000 nM T98896 CUE3W5 44425399 IC50 = 10000 nM T98896 CAK1Y9 44425400 IC50 = 9200 nM T98896 COS8W2 44425401 IC50 = 6800 nM T98896 CU74SP 44425402 IC50 > 67000 nM T98896 C7VY4P 44425403 IC50 > 67000 nM T98896 C51LRU 44425404 IC50 > 67000 nM T98896 CCI0Z9 44425405 IC50 > 22000 nM T98896 C6J1OI 44425406 IC50 > 67000 nM T98896 CK5FX1 44425407 IC50 > 67000 nM T98896 C05UME 44425408 IC50 > 67000 nM T98896 C5BH6C 44425409 IC50 > 67000 nM T98896 CF2J7B 44425410 IC50 = 900 nM T98896 CA1C5R 44425411 IC50 = 1100 nM T98896 CRT7C6 44425412 IC50 = 1300 nM T98896 C6R3OW 44425413 IC50 = 11100 nM T98896 CW8NS0 44425414 IC50 = 1300 nM T98896 C1TL9O 44425415 IC50 = 1600 nM T98896 C2GE8F 44425416 IC50 = 1800 nM T98896 CDE9I0 44432462 IC50 = 23200 nM T98896 C4NK7V 44432463 IC50 = 2200 nM T98896 C75YLA 44432466 IC50 = 2500 nM T98896 CRW6N3 44432467 IC50 = 4200 nM T98896 CV43LN 44432468 IC50 = 9000 nM T98896 C6O2RN 44432469 IC50 = 2100 nM T98896 C2VW8F 44432478 IC50 = 3700 nM T98896 CTWF60 44432479 IC50 = 6700 nM T98896 CT8FI0 44432480 IC50 = 4600 nM T98896 C98YIE 44432482 IC50 = 16900 nM T98896 CQX72A 44432483 IC50 = 14100 nM T98896 CR5D3N 44432484 IC50 = 8300 nM T98896 CAC73T 44432485 IC50 = 8000 nM T98896 CQCF94 44432486 IC50 = 11700 nM T98896 CK9MB3 44432487 IC50 = 4600 nM T98896 CQ1X5C 44432518 IC50 = 4200 nM T98896 C4XZN2 44432520 IC50 = 7100 nM T98896 COHQ74 44432521 IC50 = 9100 nM T98896 C0MHR1 44571371 IC50 = 4840 nM T98896 CTS2K7 44571372 IC50 = 1350 nM T98896 CP31DR 44571465 IC50 = 620 nM T98896 C43IBX 44571592 IC50 = 940 nM T98896 C47XUD 44571675 IC50 = 940 nM T98896 CGN2V3 44571839 IC50 = 1020 nM T98896 CJ83YR 44580388 IC50 = 37000 nM T98896 CZ5J6U 44580389 IC50 = 2600 nM T98896 C63ZCN 44580390 IC50 > 100000 nM T98896 C0ESB2 44582139 IC50 = 170 nM T98896 CWK05A 44582164 IC50 = 750 nM T98896 CDF6W8 44582402 IC50 = 1100 nM T98896 C0IEU3 44582403 IC50 = 6600 nM T98896 C3K8TQ 44582432 IC50 = 820 nM T98896 CF1AT2 44582433 IC50 = 320 nM T98896 C06CZU 44582434 IC50 = 180 nM T98896 CEG76I 44582467 IC50 = 190 nM T98896 CE4HL2 44582468 IC50 = 73 nM T98896 C4Z1VL 44582469 IC50 = 230 nM T98896 CSX5I9 46175170 IC50 = 7.4 nM T98896 C9XQZ2 46845568 IC50 = 950 nM T98896 C7IXV6 46849757 IC50 > 10000 nM T98896 C1SMH8 46882594 IC50 = 210 nM T98896 CKS5U3 46882632 IC50 = 60 nM T98896 CE9A4U 46882633 IC50 = 94 nM T98896 CUSM82 46882635 IC50 = 100 nM T98896 C5XD4Z 46882636 IC50 = 80 nM T98896 CPK4X6 46882678 IC50 = 10 nM T98896 C4VEZ3 46882679 IC50 = 21 nM T98896 C7HTW4 46882680 IC50 = 120 nM T98896 CN4J9V 46882681 IC50 = 32 nM T98896 CPD5Q4 46882720 IC50 = 770 nM T98896 C4NZL1 46882721 IC50 = 360 nM T98896 CJ8B9Y 46882762 IC50 = 800 nM T98896 C14PIN 49831179 IC50 = 6000 nM T98896 CUD7O0 50941549 IC50 = 8.4 nM T98896 CXF4V3 50990921 IC50 = 23 nM T98896 C41WIZ 52940878 IC50 > 100000 nM T98896 CV0T8G 52942214 IC50 > 100000 nM T98896 CQRD08 52942249 IC50 > 100000 nM T98896 C5P7NX 52942284 IC50 = 13000 nM T98896 CYJK29 52942928 IC50 > 100000 nM T98896 CM6X3V 52943338 IC50 = 22000 nM T98896 C7ZBC8 52943340 IC50 > 100000 nM T98896 C6PG8J 52943404 IC50 = 27000 nM T98896 CK23AZ 52944638 IC50 > 100000 nM T98896 C6U2CK 52945850 IC50 = 13000 nM T98896 C59XCQ 52945886 IC50 > 100000 nM T98896 C7CV6M 52947039 IC50 = 47000 nM T98896 C5BY4E 52947041 IC50 = 22000 nM T98896 C28MDL 52947079 IC50 = 11000 nM T98896 CQXJ52 52948198 IC50 > 100000 nM T98896 C4MK6F 52949371 IC50 > 100000 nM T98896 CXF12J 52949453 IC50 = 38000 nM T98896 CC41LX 52949467 IC50 > 100000 nM T98896 C1Y5UN 52951473 IC50 = 92 nM T98896 CXYJ67 52951474 IC50 = 270 nM T98896 C8J9EM 52951589 IC50 = 60 nM T98896 CEAS70 52951591 IC50 = 20 nM T98896 C4DG1F 52951593 IC50 = 100 nM T98896 C6XJ3V 52951596 IC50 = 250 nM T98896 C9U3AF 52951710 IC50 = 66 nM T98896 C4M1CA 52951712 IC50 = 330 nM T98896 CGC83H 52951843 IC50 > 1000 nM T98896 C76LDY 52951967 IC50 = 17 nM T98896 CYKS94 52951968 IC50 = 19 nM T98896 CE0FP3 52951969 IC50 = 23 nM T98896 CL69OM 52951970 IC50 = 29 nM T98896 CMPB74 52951971 IC50 = 2.9 nM T98896 CZ1TN8 52951972 IC50 = 8.3 nM T98896 CK08OB 52952074 IC50 = 10 nM T98896 C46AYR 52952075 IC50 = 87 nM T98896 CR32ZW 52952076 IC50 = 62 nM T98896 CJ9O3S 52952077 IC50 = 37 nM T98896 C3N9TF 52952078 IC50 = 47 nM T98896 C5S1IG 52952079 IC50 = 410 nM T98896 CKV9R0 52952178 IC50 = 330 nM T98896 CV0R6Y 52952179 IC50 = 230 nM T98896 CE4Q7F 52952273 IC50 = 180 nM T98896 CMA69V 52952274 IC50 = 33 nM T98896 C7KB5W 52952275 IC50 = 27 nM T98896 CRO0X4 52952276 IC50 = 130 nM T98896 CSJ05E 52952277 IC50 = 67 nM T98896 C29UJB 52952388 IC50 = 39 nM T98896 C3H5ID 52952389 IC50 = 21 nM T98896 CSX69R 52952390 IC50 = 110 nM T98896 CB36KP 52952492 IC50 = 320 nM T98896 C67OEU 52952493 IC50 = 17 nM T98896 CV1I0A 52952597 IC50 = 8.6 nM T98896 CGI87K 52952598 IC50 = 38 nM T98896 CXWI18 52952599 IC50 = 14 nM T98896 C46VHP 52952600 IC50 = 10 nM T98896 CH3G6R 52952601 IC50 = 29 nM T98896 CC0Y3M 52952602 IC50 = 17 nM T98896 CMQZ70 53242178 IC50 = 860 nM T98896 CSUW40 54352406 IC50 = 1410 nM T98896 C3M8GZ 54580051 IC50 = 3400 nM T98896 CL0WM9 54580052 IC50 = 480 nM T98896 CK26XF 54580053 IC50 = 1500 nM T98896 CA6K5D 54581029 IC50 = 11 nM T98896 CVK72M 54582073 IC50 = 69 nM T98896 CBK18O 54582074 IC50 = 1500 nM T98896 CP2F1B 54582075 IC50 = 250 nM T98896 CZNU23 54582076 IC50 = 1200 nM T98896 C0U5HZ 54582077 IC50 = 850 nM T98896 C8SG9Y 54582079 IC50 = 950 nM T98896 CZI6S3 54582080 IC50 = 630 nM T98896 CY50KX 54582081 IC50 = 79 nM T98896 CH6Q2Z 54583016 IC50 = 270 nM T98896 C3V9LQ 54583017 IC50 = 1700 nM T98896 CT80KQ 54583018 IC50 = 31 nM T98896 CPT4L5 54583019 IC50 = 5200 nM T98896 CBEV27 54584024 IC50 = 530 nM T98896 CM87DP 54584025 IC50 = 580 nM T98896 C3JY9Z 54584969 IC50 = 13 nM T98896 CBJ5U9 54584970 IC50 = 61 nM T98896 C28GKQ 54585927 IC50 = 450 nM T98896 CAZ76E 54586892 IC50 = 310 nM T98896 CM0OQ3 54586893 IC50 = 270 nM T98896 CK1NS7 54586894 IC50 = 410 nM T98896 CMC4Y1 54586895 IC50 = 820 nM T98896 C2MKX5 54586896 IC50 = 5400 nM T98896 CU91QP 54586897 IC50 = 1900 nM T98896 CI08RQ 54586898 IC50 = 65 nM T98896 C6PRI4 54586899 IC50 = 1400 nM T98896 C9UJ8H 54586903 IC50 = 1100 nM T98896 CKR9V8 56659819 IC50 = 4300 nM T98896 CL0U6N 56663282 IC50 = 57300 nM T98896 CI80OC 56670131 IC50 = 800 nM T98896 CO2NY6 56670132 IC50 = 24300 nM T98896 CK47BT 56928417 IC50 = 2380 nM T98896 C60GEH 66559338 IC50 > 10000 nM T98896 CF17AV 66559340 IC50 > 10000 nM T98896 C4E2BL 66559341 IC50 > 10000 nM T98896 C9I0XJ 66559342 IC50 = 6500 nM T98896 CPGK53 66559416 IC50 = 5800 nM T98896 CM7WR2 66559420 IC50 > 10000 nM T98896 CC2M8V 66559498 IC50 > 10000 nM T98896 C5QCV1 66559499 IC50 = 50 nM T98896 CCK4H3 66559500 IC50 = 230 nM T98896 C9PQ5B 66559501 IC50 > 10000 nM T98896 CG0KR4 66559502 IC50 = 460 nM T98896 CY3A5S 66559578 IC50 = 700 nM T98896 C70DOC 66559579 IC50 = 720 nM T98896 CSX64J 66559580 IC50 = 1250 nM T98896 CPB92X 66559581 IC50 = 5300 nM T98896 CP46ZL 66559668 IC50 = 1800 nM T98896 C8H7KC 66559669 IC50 = 4100 nM T98896 CS9KX1 66559670 IC50 = 1500 nM T98896 CWNJ28 66559671 IC50 = 1600 nM T98896 C57GJW 66559672 IC50 = 2600 nM T98896 C52ESR 66559934 IC50 = 50 nM T98896 C57ARI 66560021 IC50 = 30 nM T98896 CU58DB 66560022 IC50 = 40 nM T98896 CZ4E9J 66560023 IC50 > 10000 nM T98896 CI59KC 66560024 IC50 > 10000 nM T98896 CEB70Q 66560114 IC50 = 1560 nM T98896 CQ9KL4 66560115 IC50 > 10000 nM T98896 CD6R1E 66560116 IC50 > 10000 nM T98896 CGSX23 66560215 IC50 = 240 nM T98896 CIZW45 66560216 IC50 = 110 nM T98896 C3QEU0 66560217 IC50 = 390 nM T98896 CBV43Y 66560300 IC50 = 3500 nM T98896 CG98VZ 66560301 IC50 = 50 nM T98896 C4VFA8 66560302 IC50 > 10000 nM T98896 CNI8L2 66560387 IC50 = 120 nM T98896 C92GSF 66560388 IC50 = 3800 nM T98896 C16RDM 66560389 IC50 = 70 nM T98896 CM04ID 66560390 IC50 = 1600 nM T98896 C8RZG9 66560479 IC50 = 90 nM T98896 CWYS30 66560480 IC50 = 260 nM T98896 CL1Q3K 66560481 IC50 = 210 nM T98896 CA83EQ 66560482 IC50 = 2140 nM T98896 CX1MA5 66560561 IC50 = 60 nM T98896 CB8MN7 66560562 IC50 > 10000 nM T98896 C2J5GR 66560563 IC50 > 10000 nM T98896 C7C5OW 66560564 IC50 = 430 nM T98896 C9M7AN 66560645 IC50 = 870 nM T98896 CO3FU8 66560646 IC50 = 1170 nM T98896 C7S4ZM 66560647 IC50 > 10000 nM T98896 CXL86S 66560648 IC50 = 4100 nM T98896 CJO4U6 66560649 IC50 = 410 nM T98896 CKW2Q5 71453375 IC50 = 30 nM T98896 C4EJS0 71579827 IC50 = 2800 nM T98896 CO2DN4 71579916 IC50 = 2900 nM T98896 C5YF0B 71579917 IC50 = 4200 nM T98896 CNX9B1 71652215 IC50 = 1770 nM T98896 C7RZN9 71652216 IC50 = 620 nM T98896 C0NTU7 71652382 IC50 = 3500 nM T98896 CA5XS1 71652383 IC50 = 35 nM T98896 CGQK53 73346500 IC50 = 670 nM T98896 CUK6A4 73346501 IC50 > 100000 nM T98896 CNE5R7 73346502 IC50 = 340 nM T98896 CMO17L 73346503 IC50 = 880 nM T98896 CNXZ21 73346504 IC50 > 100000 nM T98896 CVM05U 73346505 IC50 = 1000 nM T98896 CUD0N8 73346506 IC50 = 100000 nM T98896 C4P5IE 73346507 IC50 = 10000 nM T98896 CY1UX5 73347990 IC50 > 100000 nM T98896 C2SPW8 73347991 IC50 = 60000 nM T98896 CW0FP6 73347992 IC50 = 1000 nM T98896 CP8M5V 73347993 IC50 = 1700 nM T98896 C4AK7S 73347994 IC50 = 1700 nM T98896 CB1R2H 73349533 IC50 > 100000 nM T98896 CADE65 73349534 IC50 = 1260 nM T98896 CW01EA 73349535 IC50 = 170 nM T98896 CE79UD 73349536 IC50 = 490 nM T98896 C02XCS 73349537 IC50 = 2300 nM T98896 CI63PO 73351092 IC50 = 300 nM T98896 CO9WP7 73351093 IC50 > 100000 nM T98896 CB09UJ 73351094 IC50 = 1600 nM T98896 CK3NC5 73351095 IC50 = 1200 nM T98896 C82OGI 73352555 IC50 = 1100 nM T98896 CR8QC6 73352556 IC50 > 100000 nM T98896 CK8U6F 73352557 IC50 = 1400 nM T98896 C73VFD 73352558 IC50 = 3200 nM T98896 C4PLA5 73354043 IC50 = 1600 nM T98896 CBZE87 73354044 IC50 = 540 nM T98896 C8VHE5 73354045 IC50 = 6300 nM T98896 C75IRY 73354046 IC50 = 700 nM T98896 CV2HI1 73354047 IC50 = 6900 nM T98896 C6KT7N 73354048 IC50 = 4100 nM T98896 C3M5QH 73354049 IC50 = 1200 nM T98896 C8WC1K 73355580 IC50 = 810 nM T98896 CNB81I 73355581 IC50 = 2100 nM T98896 C8G4FB 73357121 IC50 = 8700 nM T98896 CFZ3U6 73357122 IC50 = 5200 nM T98896 CL3CN8 73357123 IC50 > 100000 nM T98896 C5TMC1 73357124 IC50 = 3100 nM T98896 C1K5AJ 73357125 IC50 = 3300 nM T98896 CZ4VT3 73357126 IC50 = 4000 nM T98896 C3GH4V 73357127 IC50 = 1900 nM T98896 CX2NY3 73357128 IC50 = 100000 nM T98896 CB53YU 73357129 IC50 = 1200 nM T98896 CA5T7P 73603957 IC50 = 2 nM T98896 C8VN1R 74221194 IC50 = 1 nM T98896 C9HLA6 76313864 IC50 = 5000 nM T98896 CTW5H3 76317387 IC50 = 1400 nM T98896 CBQ8S2 76328307 IC50 = 6000 nM T98896 CUE7G4 86287514 IC50 = 350 nM T98896 CGQ8F3 86287515 IC50 = 17 nM T98896 CJ37XE 86287516 IC50 = 9 nM T98896 CO2FL5 90137145 IC50 = 5 nM T98896 CRT54C 101910871 IC50 = 4 nM T98896 C6VD3T 118722685 IC50 = 150 nM T98896 C5ZS4E 118722686 IC50 = 22 nM T98896 CIZB24 118722687 IC50 = 19 nM T98896 C5C0ZX 118722688 IC50 = 19 nM T98896 CTN42D 132941363 IC50 = 4 nM T98896 CAUE70 135399634 IC50 = 5400 nM T98896 CHZ03B 135722677 IC50 = 470 nM T98896 CH9SQ0 135753731 IC50 = 1300 nM T98896 CICV84 136219121 IC50 = 2200 nM T98896 CEJ8K5 136219122 IC50 = 1400 nM T98896 C4QZD7 136219123 IC50 = 830 nM T98896 C1OVE5 136219124 IC50 = 1200 nM T98896 C7F8PQ 136219125 IC50 = 1200 nM T98896 C51ULF 136219126 IC50 = 7000 nM T98896 C4PF2K 136219127 IC50 = 840 nM T98896 CZYN47 136219128 IC50 = 400 nM T98896 CABW97 136219129 IC50 = 470 nM T98896 CNF51Q 136219130 IC50 = 3000 nM T98896 C4O1PA 136219131 IC50 = 4000 nM T98896 C9GQC7 136219132 IC50 = 430 nM T98896 C6F5ZR 136219133 IC50 = 1000 nM T98896 C1CFA2 136219134 IC50 = 720 nM T98896 CAT0I7 136219135 IC50 = 6400 nM T98896 CJG54U 136219136 IC50 = 1200 nM T98896 C7U4TR 136219137 IC50 = 500 nM T98896 C28DPJ 136219138 IC50 = 420 nM T98896 C49HAE 136219139 IC50 = 730 nM T98896 CK0N4U 136219140 IC50 = 1200 nM T98896 C3CAV5 136219141 IC50 = 230 nM T98896 C6V7WB 136219142 IC50 = 630 nM T98896 C5N7MS 136219143 IC50 = 420 nM T98896 C0MA6G 136219144 IC50 = 430 nM T98896 CDG15I 136224204 IC50 = 2500 nM T98896 C8I4MK 136224205 IC50 = 1700 nM T98896 CK5J6H 136228184 IC50 = 5300 nM T98896 CBE94M 136240106 IC50 = 480 nM T98896 CIWC65 136240282 IC50 = 480 nM T98896 CPN1G2 136240283 IC50 = 420 nM T98896 C8T5IM 136241628 IC50 = 2700 nM T98896 C9RQ8K 136241629 IC50 = 6000 nM T98896 CPB07Z 136241630 IC50 = 170 nM T98896 COJ2Y9 136241631 IC50 = 410 nM T98896 CLBH50 136241632 IC50 = 4000 nM T98896 CTN9J8 136245081 IC50 = 500 nM T98896 CM2QF6 136245082 IC50 = 500 nM T98896 C75CQR 136245083 IC50 = 1300 nM T98896 C3LWO9 136249364 IC50 = 1700 nM T98896 CTD06C 136249365 IC50 = 430 nM T98896 CBPV78 136249366 IC50 = 1400 nM T98896 CWK7U9 136249367 IC50 = 380 nM T98896 CF4YX2 136249368 IC50 = 470 nM T98896 CAE17Z 136249369 IC50 = 700 nM T98896 C5XYP2 136264448 IC50 = 1500 nM T98896 C9GOS5 136264449 IC50 = 1700 nM T98896 CS80YI 137652598 IC50 = 13 nM T98896 CZ8H6N 137661550 IC50 = 5 nM T98896 CZ25LW 155512044 IC50 = 3 nM T98896 CP9YX2 155567218 IC50 = 110 nM T98896 C8D5VK 155567855 IC50 = 9 nM T98896 D0FD9M 54585928 IC50 = 20 nM T98896 D0H6CK 10160968 Ki = 97 nM T92185 CE0YO6 9824797 Ki = 604 nM T92185 C1UX9C 9955419 Ki = 72 nM T92185 CGEJ24 9985625 IC50 > 7000 nM T92185 C4CST7 24868185 IC50 = 56.7 nM T92185 CYI8C2 25022641 Ki = 85 nM T92185 CCB52N 25022642 Ki = 185 nM T92185 CTLA59 25022654 Ki = 204 nM T92185 CZQS64 25022655 Ki = 140 nM T92185 C5UB1A 25022656 Ki = 274 nM T92185 C4GJ1T 25022657 Ki = 241 nM T92185 CVD12P 44373782 Ki = 56 nM T92185 CO57KW 44453683 Ki = 404 nM T92185 CPHI72 44453791 Ki = 152 nM T92185 CFIS06 44453792 Ki = 167 nM T92185 C3XOU1 44453861 Ki = 554 nM T92185 CHQ5O6 44454004 Ki = 537 nM T92185 CZ98NW 44454024 Ki = 522 nM T92185 CS7H1K 44566176 EC50 = 49.4 nM T92185 CT4Z1R 127034614 IC50 = 53 nM T92185 CU12JI 127035881 IC50 = 57 nM T53952 D0E3TC 44259 IC50 = 585 nM T53952 D03BNU 59604787 IC50 > 10000 nM T53952 CLS29B 46872626 IC50 > 10000 nM T53952 CDK93W 56946894 IC50 = 40 nM T53952 C8X5JG 57384039 IC50 = 30 nM T53952 CV63UL 67240318 IC50 > 10000 nM T53952 C4TM6F 70682212 IC50 < 3 nM T53952 C9PE4T 70682214 IC50 = 570 nM T53952 CW4C1K 70684312 IC50 = 20 nM T53952 C7OX5Z 70686473 IC50 = 50 nM T53952 CP08FT 70696865 IC50 = 60 nM T53952 CJ2T9E 76332983 IC50 > 10000 nM T53952 C4Q5LF 132471857 IC50 < 3 nM T53952 C3TS2A 132968992 IC50 = 30 nM T53952 CY36QB 136254272 IC50 < 3 nM T53952 C2MD1Q 155513187 IC50 > 10000 nM T53952 D00ERW 44444843 Ki > 3338 nM T53952 D04TPA 72163809 IC50 = 40 nM T53952 D0L4WN 31420 IC50 = 3300 nM T52450 D00MDP 466151 IC50 = 4.9 nM T52450 D05VZE 119031 Ki = 0.7 nM T52450 D0HG5M 11452716 IC50 = 33 nM T52450 D0MW3H 9824350 Ki = 0.3 nM T52450 D0N4IV 10718956 IC50 > 1000 nM T52450 D09EFW 46861776 IC50 = 5319.54 nM T52450 D00UCC 9827497 IC50 = 8900 nM T52450 D01DVX 9847838 IC50 = 429 nM T52450 D03BOZ 3342298 IC50 = 34 nM T52450 D05VNG 9908389 IC50 = 2.2 nM T52450 D08CEE 10478364 Ki = 760 nM T52450 D0E5GY 9904965 Ki = 2 nM T52450 D0EF7V 5487313 IC50 = 40 nM T52450 D0H5CD 5748217 IC50 = 20 nM T52450 D0P8YC 5362422 Ki = 0.5 nM T52450 D0Q1CD 6918336 Ki = 5000 nM T52450 D0T2IQ 443600 IC50 = 1100 nM T52450 D0T9HG 132519 IC50 = 0.2 nM T52450 D0Y1XT 128564 Ki < 1 nM T52450 CNA81R 1836 IC50 > 2000 nM T52450 CY78XM 4218 Ki = 24 nM T52450 CZ45IU 4219 IC50 = 4.1 nM T52450 CFY8Q2 4230 IC50 = 24 nM T52450 C9EW1B 4369 Ki = 23 nM T52450 C3JZ6K 5111 Ki = 70 nM T52450 CL15AQ 65373 IC50 = 50120 nM T52450 CYEU83 69033 Ki = 79000 nM T52450 C0PY5N 77754 Ki > 100 nM T52450 CP4O2C 121255 Ki = 71000 nM T52450 CXO86G 154135 IC50 = 4650 nM T52450 CDJS43 154136 IC50 = 79 nM T52450 C50IPY 154137 IC50 = 51 nM T52450 C7ROG5 177347 IC50 > 10000 nM T52450 CP7Q8T 240910 Ki = 34000 nM T52450 CX3DK6 283995 Ki = 29000 nM T52450 COFX01 352863 Ki = 71000 nM T52450 CV60YH 445010 IC50 = 212 nM T52450 CK9M3P 445018 IC50 = 22.2 nM T52450 C4D7TS 448002 Ki = 174 nM T52450 CR51PG 448593 Ki = 470 nM T52450 C9I8WB 478379 Ki = 0.1 nM T52450 C45JSH 639942 IC50 = 5403.64 nM T52450 CP91NX 677915 IC50 = 3451.32 nM T52450 CDE9V2 689424 IC50 = 4585.74 nM T52450 C5O0TJ 690158 IC50 = 3057.91 nM T52450 C7TPR6 690965 IC50 = 5301.68 nM T52450 CP1Q6R 703233 IC50 = 114000 nM T52450 C9FL2X 721434 IC50 = 5393.29 nM T52450 CTO15S 727131 IC50 = 4261.69 nM T52450 CTV50K 727184 IC50 = 4194.94 nM T52450 C2CL6X 732134 IC50 = 5182.87 nM T52450 CPKI76 765318 IC50 = 3159.54 nM T52450 CXME85 766168 IC50 = 3501.61 nM T52450 CQB03J 780790 IC50 = 4515.39 nM T52450 C7EHR1 787183 IC50 = 4670.92 nM T52450 C5MF2E 795596 IC50 = 5255.29 nM T52450 C1K0NF 795855 IC50 = 3252.67 nM T52450 CW56XG 875024 IC50 = 4173.64 nM T52450 C17IXT 910211 IC50 = 3303.83 nM T52450 C9IFC6 1348435 IC50 = 93000 nM T52450 CN9C8D 2140735 IC50 = 860000 nM T52450 CN6E3U 2366268 IC50 > 10000 nM T52450 CN62WX 2800809 IC50 = 7000 nM T52450 CY3TD6 3348132 Ki > 2000 nM T52450 CME24U 3649035 IC50 > 101000 nM T52450 C3EI6T 4085085 IC50 = 400000 nM T52450 CC5O4E 4369384 IC50 = 2200 nM T52450 CP8D7Y 4478236 IC50 = 6150 nM T52450 CZBY34 5220706 Ki = 66000 nM T52450 C20HRJ 5273475 IC50 = 5201.56 nM T52450 CH01XT 5281656 IC50 = 11360 nM T52450 CQ4VL5 5287415 IC50 = 1300 nM T52450 CW5SE3 5288615 IC50 = 6.6 nM T52450 CJ3QI1 5288814 IC50 = 7780 nM T52450 C5IDT0 5289314 Ki = 25 nM T52450 CO58XD 5311161 IC50 > 100000 nM T52450 CVLS16 5319161 IC50 = 16320 nM T52450 CL89FO 5496920 Ki = 303 nM T52450 CDI23X 5941957 IC50 > 100000 nM T52450 C5OMB7 6102708 IC50 = 97 nM T52450 C0M3LR 6323382 IC50 = 7 nM T52450 CL5DH0 6479915 IC50 = 14700 nM T52450 CI86PQ 6539651 IC50 = 170 nM T52450 CQEF36 6539670 IC50 = 50 nM T52450 CP7BG0 6852146 IC50 > 16000 nM T52450 CN5L2B 6852147 IC50 = 150 nM T52450 CP2XK7 6882342 IC50 = 360000 nM T52450 CPFV65 6916013 Ki > 200 nM T52450 C57XJO 7550925 IC50 = 55000 nM T52450 C7Y1BX 9543420 IC50 = 20.5 nM T52450 C9UPD8 9794928 IC50 = 8040 nM T52450 CIJ25V 9794947 IC50 = 80000 nM T52450 CLK61C 9797144 Ki = 82 nM T52450 CA0ZH1 9798114 IC50 = 2454.71 nM T52450 C7NP9Z 9798247 IC50 = 5450 nM T52450 C78EKW 9798637 IC50 = 676 nM T52450 C5RDZ4 9799316 IC50 = 17 nM T52450 C80WFI 9800763 IC50 = 200 nM T52450 CET56A 9801414 Ki = 2000 nM T52450 C76RCQ 9801569 IC50 = 4670 nM T52450 C68HMJ 9801786 IC50 > 10000 nM T52450 CM9GH8 9802180 IC50 = 18 nM T52450 CJY12B 9802219 Ki > 5000 nM T52450 C4CN0H 9802436 Ki = 5.3 nM T52450 CIXD67 9802768 IC50 = 8660 nM T52450 C40THQ 9802812 IC50 = 15000 nM T52450 C83FVW 9803207 IC50 = 1720 nM T52450 C3QS5H 9803407 IC50 = 2637 nM T52450 CUSD58 9803469 IC50 > 10000 nM T52450 C4QCG9 9803771 IC50 = 61 nM T52450 C23VTC 9804342 IC50 = 1600 nM T52450 C49HNU 9805016 IC50 = 1500 nM T52450 CP65QD 9805079 Ki > 5000 nM T52450 CXSU10 9805304 IC50 = 3203 nM T52450 CO4D0U 9805473 IC50 = 20 nM T52450 C1HP7E 9805710 IC50 = 9500 nM T52450 CT8X1F 9806970 IC50 = 3815 nM T52450 C76CKA 9807105 Ki > 5000 nM T52450 CTK6J8 9808181 IC50 > 100000 nM T52450 C67XKV 9808391 IC50 = 115 nM T52450 CS07BM 9808594 IC50 = 75 nM T52450 C9RQM7 9808674 IC50 > 10000 nM T52450 CTO36D 9817594 IC50 > 100000 nM T52450 C32ODL 9818295 IC50 = 6430 nM T52450 C0R2KN 9818588 IC50 > 10000 nM T52450 CC9VY4 9819420 IC50 = 3680 nM T52450 C1VT4J 9819974 IC50 = 162 nM T52450 CQG86S 9820708 IC50 = 3420 nM T52450 C6KJ9W 9822461 IC50 = 77 nM T52450 C6IX7G 9822926 IC50 = 435 nM T52450 C1MPW9 9823182 IC50 > 2000 nM T52450 CTF8V4 9823391 Ki > 5000 nM T52450 CY1H0O 9824331 IC50 = 2200 nM T52450 CUZ25T 9825237 IC50 = 870.96 nM T52450 CT6OZ1 9825650 EC50 = 15.9 nM T52450 C3AEF4 9825692 IC50 = 4730 nM T52450 CDJB86 9825720 IC50 = 74 nM T52450 CXL65P 9825920 Ki > 4900 nM T52450 CL0G8K 9825927 IC50 = 80 nM T52450 C65ZHY 9826199 IC50 = 50000 nM T52450 CVSJ72 9826275 IC50 = 2610 nM T52450 C1I6KQ 9826286 Ki > 10000 nM T52450 C7W3TG 9826481 IC50 = 1228 nM T52450 CPW60S 9827023 IC50 = 260 nM T52450 C3SZ8Y 9827469 Ki > 5000 nM T52450 C24CZI 9827635 IC50 = 125 nM T52450 C2TU0C 9827807 IC50 = 55 nM T52450 CL59JS 9827846 IC50 = 34 nM T52450 C7I2FO 9828039 Ki = 788 nM T52450 C1GR4N 9828276 IC50 > 25000 nM T52450 C7SRM4 9837496 IC50 = 100 nM T52450 C8WH1Q 9840355 IC50 = 239 nM T52450 CU7FM2 9840390 IC50 = 5110 nM T52450 CEAZ87 9840395 IC50 = 4948 nM T52450 CKF84D 9840581 IC50 = 11 nM T52450 C9PW7L 9841168 Ki > 4949 nM T52450 C5XL7R 9841323 IC50 = 170 nM T52450 CA7DJ9 9842114 IC50 = 4400 nM T52450 CQ5L0D 9842167 IC50 > 10000 nM T52450 CH63ZI 9842332 IC50 = 148 nM T52450 C6YT5W 9843479 IC50 > 10000 nM T52450 C9N5PA 9843679 IC50 = 740 nM T52450 C49UOA 9844245 IC50 = 5400 nM T52450 CK76RW 9845271 IC50 = 2640 nM T52450 C4RNT6 9845430 IC50 = 11 nM T52450 CEB90C 9846418 IC50 = 2380 nM T52450 C8T0BQ 9846437 IC50 = 398 nM T52450 CWY1J9 9846501 Ki > 5000 nM T52450 C4D2MY 9846507 IC50 = 662 nM T52450 CI7T1S 9846676 IC50 = 220 nM T52450 C0KP9H 9847092 IC50 = 2560 nM T52450 CE9AL3 9847113 IC50 = 1140 nM T52450 CA1IP0 9847191 Ki > 5000 nM T52450 C8IMT2 9847787 IC50 = 1.1 nM T52450 C6SV1X 9847843 IC50 = 238 nM T52450 C7VXJ5 9848025 IC50 = 9.1 nM T52450 CG14CO 9848625 IC50 = 2364 nM T52450 C92EJW 9849379 IC50 = 3670 nM T52450 CX3EW2 9849576 IC50 = 3372 nM T52450 CHVL24 9849957 IC50 = 393 nM T52450 C4IEK0 9850035 IC50 > 10000 nM T52450 C9P1BH 9851086 IC50 = 1950 nM T52450 CD1KW6 9851858 Ki = 385 nM T52450 C5DGI9 9851911 IC50 = 1200 nM T52450 C2FYO3 9852206 Ki = 302 nM T52450 C7UP3K 9857957 IC50 = 220 nM T52450 CC70WV 9858468 IC50 = 5141 nM T52450 CECR39 9860227 IC50 > 30000 nM T52450 CR37HQ 9861014 IC50 ~ 10000 nM T52450 C5TUJ7 9862317 IC50 = 1560 nM T52450 C8CEJ4 9862349 IC50 = 11 nM T52450 C8GE7U 9862764 IC50 > 2000 nM T52450 CS5JT6 9864502 IC50 = 12700 nM T52450 CGUF07 9865358 IC50 = 12000 nM T52450 CU51IV 9865936 IC50 = 492 nM T52450 CI8Z0R 9866250 IC50 = 420 nM T52450 CM97TO 9866534 IC50 > 1000 nM T52450 CR10NL 9866770 Ki > 5000 nM T52450 CP4Y7O 9867411 IC50 = 96 nM T52450 C0YN1X 9867935 IC50 = 3250 nM T52450 CK3F1T 9868079 IC50 > 10000 nM T52450 CX57RB 9868249 Ki > 5000 nM T52450 C2L9SU 9868329 IC50 = 34 nM T52450 CJS23I 9868333 Ki > 4949 nM T52450 C5O0GC 9868490 IC50 = 1752 nM T52450 CRI23M 9868515 IC50 = 113 nM T52450 C4K2GH 9868577 IC50 = 368 nM T52450 C4ZR7O 9868713 IC50 = 835 nM T52450 C24JSB 9868858 IC50 > 10000 nM T52450 C5IJH2 9869068 IC50 = 318 nM T52450 CT76IN 9869441 IC50 = 450 nM T52450 CLQ29X 9869597 IC50 = 3230 nM T52450 CA6G0W 9869598 IC50 = 2900 nM T52450 CG17NZ 9869811 IC50 = 4600 nM T52450 CZO6K4 9869819 IC50 = 16 nM T52450 C5ELS6 9869902 IC50 = 598 nM T52450 CMEA71 9869947 IC50 = 2350 nM T52450 C38BVX 9870100 IC50 > 1000 nM T52450 CZO2I0 9870133 IC50 = 10000 nM T52450 CA48SX 9870269 IC50 = 67000 nM T52450 C5QFG1 9871290 IC50 = 761 nM T52450 CD1XQ2 9871305 IC50 > 50000 nM T52450 CSM16R 9871355 IC50 > 10000 nM T52450 CHU9I8 9871883 IC50 = 4000 nM T52450 C5NM6P 9872886 Ki = 5 nM T52450 CU9L3X 9879183 IC50 > 10000 nM T52450 CG41SV 9879575 IC50 > 10000 nM T52450 C0TCJ2 9880675 Ki > 4949 nM T52450 C0NA6S 9880842 IC50 = 313 nM T52450 CW8IC4 9882151 IC50 = 40000 nM T52450 C0ZT7A 9883002 Ki = 206000 nM T52450 C0QY4U 9883809 IC50 > 30000 nM T52450 C9XSN0 9883962 IC50 > 30000 nM T52450 C2OHV3 9885051 IC50 = 4440 nM T52450 CG35XZ 9885916 IC50 > 10000 nM T52450 CZBK85 9886177 IC50 > 2000 nM T52450 CCAI25 9886751 IC50 = 25 nM T52450 CHT08B 9886916 IC50 = 65 nM T52450 CJDS01 9886923 IC50 = 4320 nM T52450 C2M4EC 9887473 Ki > 4946 nM T52450 C4PB5Z 9887544 Ki = 1.2 nM T52450 C1STP9 9887771 IC50 = 290 nM T52450 CFG4Q2 9887831 IC50 = 201 nM T52450 C3ZG6O 9887870 IC50 = 6000 nM T52450 CC87LP 9888280 IC50 = 494 nM T52450 C8AJB7 9888429 Ki > 5000 nM T52450 CD76WB 9888485 IC50 = 656 nM T52450 CVP45O 9888530 IC50 = 5600 nM T52450 CJS0E5 9888649 IC50 = 158 nM T52450 CB2YG7 9889128 IC50 = 642 nM T52450 CD1U5P 9889190 IC50 = 2000 nM T52450 C4AVN6 9889449 IC50 = 475000 nM T52450 C27HMG 9889517 IC50 = 1.2 nM T52450 CZD2E3 9889870 IC50 = 1210 nM T52450 C26SZX 9890226 IC50 = 116 nM T52450 CWN19T 9890526 IC50 > 10000 nM T52450 CD79UJ 9890632 IC50 > 100000 nM T52450 CNX78A 9890733 IC50 = 1070 nM T52450 CMD0S2 9891009 IC50 = 1227 nM T52450 CN0MS4 9891048 IC50 = 15000 nM T52450 C20LGF 9891255 IC50 = 413 nM T52450 C9YD2O 9891259 IC50 = 627 nM T52450 CU65HY 9891358 IC50 > 10000 nM T52450 C3QSE6 9891814 IC50 = 3100 nM T52450 CPT4C6 9892042 IC50 = 639 nM T52450 CR50BS 9892336 IC50 = 956 nM T52450 C1KV7J 9892518 IC50 = 523 nM T52450 CH69LT 9892815 Ki > 10000 nM T52450 CZU7Y4 9892876 IC50 = 50000 nM T52450 CK1F3O 9892889 Ki > 1627 nM T52450 CSIB97 9896504 IC50 > 30000 nM T52450 C6Q4JF 9903007 IC50 = 258 nM T52450 C97GSC 9903557 Ki > 4949 nM T52450 C2R5CX 9905493 IC50 = 49 nM T52450 CD78ZQ 9907286 IC50 = 1200 nM T52450 CYHN04 9908006 IC50 = 1390 nM T52450 CMSC52 9908418 Ki > 850 nM T52450 CKWF30 9908681 IC50 = 357 nM T52450 CQ8Y9T 9909624 IC50 = 260 nM T52450 CN6WJ1 9909994 IC50 = 110 nM T52450 CVT4D1 9910032 IC50 = 30000 nM T52450 CJ3K1I 9910075 IC50 > 10000 nM T52450 CPO8V1 9910282 IC50 > 10000 nM T52450 CM2F7R 9910302 IC50 = 2.6 nM T52450 C4E6LR 9910544 IC50 = 1911 nM T52450 C6NUE9 9910550 IC50 = 31 nM T52450 CP4LS8 9910727 IC50 > 10000 nM T52450 C5IGQ1 9911009 IC50 = 1100 nM T52450 CSHR05 9911683 IC50 = 90 nM T52450 CT50EC 9912183 Ki > 5000 nM T52450 C2GMQ0 9912235 IC50 = 498 nM T52450 C62VZI 9912382 IC50 = 104 nM T52450 C8VJ9Z 9913053 IC50 = 40 nM T52450 CI5A3G 9913301 IC50 = 531 nM T52450 C3AZP0 9913479 IC50 > 10000 nM T52450 CX1Q5C 9913489 IC50 = 3790 nM T52450 CSZV76 9913881 IC50 = 25 nM T52450 C8AQ3S 9913990 IC50 = 0.88 nM T52450 C7ZY1L 9914029 IC50 = 6000 nM T52450 CU9B3E 9914147 IC50 = 124 nM T52450 C8L2IQ 9915804 Ki = 770 nM T52450 CM7UO8 9924798 IC50 = 325 nM T52450 CBPD13 9926779 IC50 = 9 nM T52450 CSA12Z 9927353 IC50 = 33 nM T52450 C4YGT6 9928325 IC50 = 3 nM T52450 C26ZPC 9929976 IC50 = 7060 nM T52450 C7EIX4 9930068 Ki = 2.8 nM T52450 CK5OV9 9930210 IC50 = 40 nM T52450 CWN0L8 9930514 IC50 = 854 nM T52450 C67PBX 9932128 IC50 = 6500 nM T52450 CJI5A7 9932167 IC50 = 1410 nM T52450 CY79AT 9932263 IC50 = 320 nM T52450 C03GVA 9932290 Ki = 400 nM T52450 C1I2FW 9932632 Ki > 5000 nM T52450 CCHZ97 9932731 IC50 = 2300 nM T52450 C3VO2E 9932958 IC50 = 29000 nM T52450 CT2KM9 9933083 IC50 = 1000 nM T52450 CDXR37 9933197 IC50 = 8000 nM T52450 C2EUL8 9933259 IC50 = 2333 nM T52450 CX17KQ 9933408 IC50 = 10300 nM T52450 C5E7PR 9933720 Ki = 1450 nM T52450 CF26MY 9934052 Ki > 5000 nM T52450 CA5V8M 9934053 Ki > 5000 nM T52450 C57WSD 9934240 IC50 > 100000 nM T52450 CGJZ78 9934997 IC50 = 841 nM T52450 C65ION 9935032 IC50 > 10000 nM T52450 CDRC76 9936405 IC50 = 4982 nM T52450 CH9G5D 9936469 IC50 = 165 nM T52450 C68MQN 9936625 Ki > 5000 nM T52450 C7GJF8 9936712 IC50 = 194 nM T52450 CG38KL 9936728 Ki = 13 nM T52450 CE59TP 9936926 IC50 > 10000 nM T52450 CX7VQ9 9937188 IC50 = 320 nM T52450 CMI06Q 9939403 Ki = 32000 nM T52450 CLM2R8 9941370 Ki = 5900 nM T52450 C0IBF2 9941371 Ki = 2440 nM T52450 C12ZGS 9945200 IC50 = 10 nM T52450 C0MLZ6 9945553 IC50 > 10000 nM T52450 CA30JY 9946988 IC50 > 10000 nM T52450 C6TH4I 9947270 IC50 > 10000 nM T52450 CSN61C 9948296 Ki > 4949 nM T52450 C16HTN 9948666 IC50 = 1895 nM T52450 C52IUJ 9949603 IC50 > 10000 nM T52450 CF1DO9 9950475 Ki > 5000 nM T52450 COVR98 9951986 IC50 = 4 nM T52450 CQY54S 9952396 IC50 = 125 nM T52450 CWO48K 9952436 IC50 = 490 nM T52450 C8C3DL 9953278 IC50 > 10000 nM T52450 C9OY4Z 9953817 IC50 = 1310 nM T52450 C16GIN 9953861 Ki > 5000 nM T52450 CR6EX3 9953909 Ki > 5000 nM T52450 CABI45 9954117 IC50 = 24 nM T52450 C8RXN6 9954304 IC50 > 10000 nM T52450 C6GA8D 9954513 IC50 = 1930 nM T52450 CH9YL3 9954604 IC50 = 629 nM T52450 C37VXK 9954605 IC50 = 519 nM T52450 C9X0YR 9954867 IC50 > 10000 nM T52450 C32HAZ 9954953 Ki = 8 nM T52450 CK9HX0 9955125 IC50 = 3600 nM T52450 CMV37W 9955127 IC50 = 3197 nM T52450 CWE6N8 9955640 IC50 = 157 nM T52450 C3ZLA1 9956465 IC50 = 2573 nM T52450 C8M2RB 9956613 IC50 > 10000 nM T52450 C3Q2UJ 9956686 IC50 = 5000 nM T52450 CS73TB 9956692 Ki > 4948 nM T52450 CI5TW9 9956699 IC50 = 14000 nM T52450 CCB6M3 9956827 IC50 = 2900 nM T52450 C56GFP 9956833 IC50 = 1330 nM T52450 CQ80MP 9957107 IC50 = 465 nM T52450 CC4WG3 9957228 Ki > 300000 nM T52450 C5I0VJ 9957500 IC50 = 7803 nM T52450 CN76XI 9957653 IC50 = 801 nM T52450 CPJR82 9957875 IC50 = 143 nM T52450 CWE4D3 9958604 IC50 = 4750 nM T52450 CVG0O2 9959014 IC50 > 1000 nM T52450 CNHT34 9959421 IC50 = 53 nM T52450 CN8TK0 9959428 IC50 > 10000 nM T52450 CV40RB 9960075 Ki > 4949 nM T52450 C9DRB7 9966028 IC50 = 28000 nM T52450 CYK75X 9967932 IC50 > 10000 nM T52450 C0HL2X 9976697 IC50 = 0.8 nM T52450 CXS48O 9979594 Ki = 14 nM T52450 CZJ8M4 9982000 IC50 = 32 nM T52450 CUA65C 9982414 IC50 = 920 nM T52450 CO09PN 9983251 IC50 = 43 nM T52450 CJGR30 9983604 IC50 = 1420 nM T52450 CILK24 9983687 Ki = 21877.62 nM T52450 C1N0MZ 9985145 Ki = 10 nM T52450 C8IL6Q 9986000 IC50 = 19 nM T52450 C3KX1B 9998685 Ki = 1085 nM T52450 CB2J3S 9999667 IC50 = 20 nM T52450 CO7Y9J 10001450 Ki = 3 nM T52450 C6TO0A 10001582 Ki = 7 nM T52450 C2D8WU 10001779 IC50 = 240 nM T52450 C59WEK 10001843 IC50 = 400 nM T52450 CM9ZV4 10002342 IC50 = 290 nM T52450 CKJB90 10002422 IC50 = 145 nM T52450 C2L3EU 10003206 Ki = 72 nM T52450 C8Q9OC 10003866 Ki = 170 nM T52450 CP5N4E 10005114 Ki = 12800 nM T52450 CVUE46 10005340 Ki = 62 nM T52450 C6U3CK 10006134 IC50 = 28.9 nM T52450 CA8C6U 10008733 Ki = 329 nM T52450 C4IFN5 10009833 IC50 = 20 nM T52450 CR7T3J 10009978 Ki > 2000 nM T52450 CJ6H8O 10019658 IC50 = 62 nM T52450 C6WHU4 10023722 IC50 = 18 nM T52450 C71YGT 10025307 Ki > 5000 nM T52450 C1N3MI 10026327 IC50 = 564 nM T52450 CEX7D8 10026420 IC50 = 39300 nM T52450 C6O0MN 10026682 Ki = 22400 nM T52450 CVCB95 10027113 IC50 = 2900 nM T52450 C6DGR7 10027203 Ki = 10 nM T52450 CY62OQ 10027598 IC50 = 27 nM T52450 C05LFQ 10028633 IC50 = 120 nM T52450 CG3BS7 10028949 IC50 = 68 nM T52450 CM52RO 10030422 IC50 = 770 nM T52450 CVG03H 10031524 IC50 = 54 nM T52450 C7J9ZF 10039403 IC50 = 3300 nM T52450 C1X0SA 10041385 Ki = 1060 nM T52450 CPZ4L1 10041481 IC50 = 14 nM T52450 CNA3G4 10042214 IC50 = 1310 nM T52450 CO39PK 10042482 Ki = 150 nM T52450 C7O8HD 10044261 IC50 = 93 nM T52450 CY1J5S 10045091 IC50 = 30 nM T52450 C7CT4E 10045150 IC50 = 21 nM T52450 CHF92V 10047100 Ki > 5000 nM T52450 CLXN48 10047373 IC50 = 490 nM T52450 CCF5Z4 10047585 IC50 = 0.3 nM T52450 CAN59F 10047708 IC50 = 1.8 nM T52450 CCA67I 10048718 Ki < 1 nM T52450 CV59KC 10049292 Ki > 10000 nM T52450 C1N9UX 10050222 IC50 = 1616 nM T52450 CZR4U6 10050655 Ki = 95 nM T52450 C19LUE 10050937 Ki = 1300 nM T52450 C1G0HE 10051959 IC50 = 270 nM T52450 CZ6R1T 10052198 Ki < 1 nM T52450 CRJ85Q 10053965 IC50 = 980 nM T52450 CSHD67 10054852 IC50 = 39 nM T52450 C42YWK 10055393 IC50 = 9120.11 nM T52450 CSW7B3 10067146 Ki = 272 nM T52450 C5KR4U 10068161 IC50 = 12 nM T52450 C5WC8A 10070323 IC50 > 10000 nM T52450 CD3RL7 10070821 Ki > 10000 nM T52450 C2P7WT 10070826 Ki = 16 nM T52450 CQ7PJ9 10072419 Ki = 30 nM T52450 CSG9A5 10073761 Ki = 1900 nM T52450 CJK0R1 10074190 IC50 = 4785 nM T52450 CV0I9M 10074738 IC50 = 87 nM T52450 CLC84V 10075168 IC50 <= 100 nM T52450 CVJ84F 10075482 IC50 = 830 nM T52450 CPS4R9 10076090 IC50 = 155 nM T52450 CR6N8D 10077348 IC50 = 23 nM T52450 CJ2H0T 10077849 IC50 = 44 nM T52450 CVTD42 10078499 Ki > 40000 nM T52450 CU7DJ1 10081163 Ki = 65000 nM T52450 CUT28D 10088847 Ki = 196 nM T52450 CPKC43 10093147 IC50 = 3245 nM T52450 C8AEK4 10093420 IC50 = 0.26 nM T52450 CK5IS6 10094143 IC50 = 520 nM T52450 CC1H2J 10094144 IC50 = 260 nM T52450 C5W4ZA 10094362 IC50 = 6 nM T52450 CHK0M7 10094867 Ki = 143 nM T52450 CA6X2Z 10095338 IC50 = 5 nM T52450 C76SQC 10097061 IC50 = 400 nM T52450 CMY3X2 10098158 IC50 = 4.8 nM T52450 C2XV5J 10098250 IC50 = 1080 nM T52450 CLF2R6 10098574 Ki = 80 nM T52450 C3V2HW 10099112 IC50 = 27000 nM T52450 CMLA47 10099961 IC50 = 38 nM T52450 CF3HQ9 10100283 Ki = 61 nM T52450 CXV2Y3 10109170 Ki > 4949 nM T52450 C0G7IY 10114318 Ki = 450 nM T52450 C9T2AW 10116042 IC50 = 111 nM T52450 CVK61T 10116047 IC50 > 1100 nM T52450 C78JHL 10116107 Ki = 430 nM T52450 C4P1LB 10116618 IC50 > 50000 nM T52450 CU0D4S 10117481 Ki > 4948 nM T52450 CP5L0W 10117663 Ki > 4900 nM T52450 CU3ZM2 10118633 IC50 > 1000 nM T52450 C2F8KW 10119294 IC50 = 933.25 nM T52450 CPA4R9 10119730 IC50 = 172 nM T52450 C7A8MI 10120093 IC50 = 4600 nM T52450 C0Q9DW 10120586 IC50 = 913 nM T52450 CT4V0P 10120622 IC50 = 2500 nM T52450 C0KHW5 10120930 IC50 = 4168.69 nM T52450 CP65KL 10125869 Ki = 213 nM T52450 CY2N3D 10127629 Ki > 4950 nM T52450 C1N4MJ 10127670 Ki > 4950 nM T52450 CIL09Z 10127889 Ki > 4950 nM T52450 C07KFI 10128313 Ki > 4950 nM T52450 CB3I6K 10128659 Ki > 4950 nM T52450 C6ZK3A 10128916 Ki > 4950 nM T52450 C35LGX 10132821 IC50 = 138 nM T52450 CS54CQ 10133565 IC50 > 10000 nM T52450 C9EWX5 10135125 IC50 = 1000 nM T52450 CDR73P 10135184 Ki > 2128 nM T52450 C7KR3Y 10136680 Ki = 460 nM T52450 CNU93J 10136924 Ki = 440 nM T52450 C1CDF2 10136925 Ki = 630 nM T52450 CJ9EX4 10138303 Ki = 1040 nM T52450 C6UXD7 10138936 IC50 = 99 nM T52450 CFXC89 10139040 Ki > 4946 nM T52450 CGC6S5 10139402 Ki > 4948 nM T52450 CP8QV4 10140363 Ki > 4948 nM T52450 CU6Y9T 10140438 Ki > 4949 nM T52450 CE75BY 10140776 Ki > 4900 nM T52450 C5DA1U 10141270 IC50 = 190.55 nM T52450 C5H1ZM 10141426 IC50 = 45.71 nM T52450 CLXF15 10141613 Ki > 4900 nM T52450 C7VF1K 10141614 Ki > 4900 nM T52450 CWB5O4 10142326 Ki > 4900 nM T52450 CL7P6G 10143019 IC50 = 6600 nM T52450 CPXB21 10143028 Ki > 4949 nM T52450 C23WZR 10143587 Ki > 4900 nM T52450 CAM6U7 10143672 IC50 = 107.15 nM T52450 C82SMW 10144091 IC50 = 100 nM T52450 CD3U8E 10150649 Ki = 25 nM T52450 CUG62E 10155007 IC50 = 14000 nM T52450 CLQ89T 10155008 IC50 = 2600 nM T52450 CZW98O 10156375 Ki > 4949 nM T52450 CPY87U 10158366 IC50 > 10000 nM T52450 CYO8D2 10159633 Ki > 4949 nM T52450 CQ4SJ5 10160197 Ki > 4948 nM T52450 CHUA34 10160545 IC50 = 7900 nM T52450 CQ41YI 10161391 Ki > 4949 nM T52450 CCU9S1 10162155 IC50 = 1805 nM T52450 C7SXD4 10162245 Ki > 4900 nM T52450 CO6PS3 10162900 Ki = 420 nM T52450 CR5H6E 10163627 Ki > 2128 nM T52450 CI9VJ5 10163857 Ki > 4948 nM T52450 CR17PV 10164205 Ki > 4948 nM T52450 CZO5V4 10164317 IC50 = 2590 nM T52450 CCM0Y8 10165180 Ki > 4900 nM T52450 CE10MK 10165419 IC50 = 172 nM T52450 CP02FJ 10165420 IC50 = 172 nM T52450 C0K7HT 10165868 IC50 = 64.57 nM T52450 C5ZO9J 10166232 IC50 > 50000 nM T52450 CNTC03 10172417 Ki = 25 nM T52450 C6IW4O 10173876 Ki > 4950 nM T52450 C4QY3V 10175210 Ki > 4950 nM T52450 C5JM1A 10179045 IC50 > 10000 nM T52450 CD4AO0 10180362 IC50 > 10000 nM T52450 CS6X2R 10183408 IC50 = 223.87 nM T52450 C6OE9H 10183692 IC50 > 10000 nM T52450 CDM94B 10183693 Ki > 4900 nM T52450 C2GV5Q 10183755 IC50 = 362 nM T52450 CHB2D3 10184071 Ki > 4948 nM T52450 CH04IS 10184457 IC50 = 39 nM T52450 C3E9NF 10184537 Ki > 4900 nM T52450 CTDP62 10184579 Ki > 4900 nM T52450 CXQ8N0 10185100 Ki > 4949 nM T52450 C2OM9G 10186288 IC50 = 3090.3 nM T52450 CK0P3F 10186536 Ki > 2128 nM T52450 CV7YI1 10186544 Ki > 4900 nM T52450 CA9FG4 10187181 IC50 = 151 nM T52450 C51RPY 10195069 Ki > 4950 nM T52450 CY36NO 10196425 Ki > 4950 nM T52450 CVRZ27 10198038 IC50 = 500 nM T52450 C0U9KC 10199401 IC50 = 672 nM T52450 C5CUM9 10202769 Ki > 4949 nM T52450 CX8BS3 10203685 Ki > 4949 nM T52450 C4FSU0 10203714 IC50 = 1400 nM T52450 CE1LI3 10204303 Ki = 360 nM T52450 C32RAQ 10204620 Ki > 4900 nM T52450 C7AU0H 10205886 IC50 = 151.36 nM T52450 CS1CA5 10207780 Ki > 4900 nM T52450 C4K1MJ 10208262 Ki > 2128 nM T52450 CYE02Q 10209301 IC50 = 50000 nM T52450 CV4DG9 10209314 IC50 = 136 nM T52450 CD76KE 10209382 Ki > 4949 nM T52450 C1C7AH 10223757 Ki > 4946 nM T52450 CYG10Z 10223774 Ki > 4948 nM T52450 C92BVJ 10223963 IC50 = 12000 nM T52450 CV5X8A 10224181 IC50 > 30000 nM T52450 CGKU70 10224396 Ki = 390 nM T52450 C7K1OR 10224602 IC50 > 10000 nM T52450 CLH71C 10225319 Ki > 4949 nM T52450 C2X1KF 10226116 Ki > 4900 nM T52450 CJ46HR 10227522 IC50 = 8.913 nM T52450 CUE63Q 10227853 Ki > 4900 nM T52450 C19DFP 10227854 Ki > 4900 nM T52450 CM7B5T 10228228 Ki > 4948 nM T52450 C7T0WH 10229644 IC50 = 1760 nM T52450 CD2HP3 10230012 Ki > 4900 nM T52450 CLJ3Y9 10230286 IC50 = 77 nM T52450 CCRM18 10231253 IC50 = 20 nM T52450 CCTY95 10237492 Ki > 4950 nM T52450 CRF32B 10237550 Ki = 23 nM T52450 CCQ9V5 10239716 Ki > 4950 nM T52450 CQ1E4F 10248274 Ki = 64 nM T52450 CLAX20 10250594 IC50 = 3.1 nM T52450 C0J3TC 10250722 Ki = 2000 nM T52450 CHGB94 10251825 Ki = 11 nM T52450 CL67DT 10252311 Ki = 548 nM T52450 CRA01T 10252319 IC50 = 2.5 nM T52450 CLX62O 10252774 Ki = 21 nM T52450 C8NS7Q 10252840 IC50 = 300 nM T52450 CK9DF5 10253223 IC50 = 2400000 nM T52450 C8LQP4 10253358 IC50 = 180 nM T52450 C2V4MP 10253549 IC50 = 71 nM T52450 CQF3V9 10253673 IC50 > 10000 nM T52450 CD8QY2 10253933 IC50 > 10000 nM T52450 CY34IB 10254279 Ki = 3 nM T52450 CJ3Q8W 10256080 IC50 = 41 nM T52450 CB6SE4 10256227 IC50 = 270 nM T52450 CP9V7O 10256251 IC50 = 280 nM T52450 CO47KX 10256290 Ki = 80 nM T52450 C8OUE9 10256513 Ki = 580 nM T52450 C4WV7B 10257654 IC50 = 152 nM T52450 CI8G0F 10258150 IC50 = 30 nM T52450 C6EI1N 10262798 Ki > 500000 nM T52450 CJKD83 10268288 IC50 > 10000 nM T52450 C0CE3N 10269452 IC50 = 1600 nM T52450 C0QS9V 10269453 IC50 = 47 nM T52450 CMNA19 10270268 IC50 > 10000 nM T52450 C2MES9 10271604 Ki = 1 nM T52450 C0K2ES 10273642 Ki > 4948 nM T52450 CJZP24 10273657 Ki > 4948 nM T52450 CK18DB 10273985 Ki > 2128 nM T52450 CGP97S 10274748 Ki = 650 nM T52450 CU67RC 10275101 IC50 = 2800 nM T52450 C13NKU 10275545 Ki > 4948 nM T52450 C1NGV9 10276473 Ki > 4948 nM T52450 CES6A5 10276821 Ki > 4900 nM T52450 C1W7SN 10277073 Ki > 4948 nM T52450 CO18TA 10277120 Ki > 4948 nM T52450 C0GU6B 10277568 IC50 = 422 nM T52450 CY6K1G 10277706 Ki > 4900 nM T52450 C9OAE1 10277812 IC50 = 550 nM T52450 C2XU3O 10278147 IC50 = 2.9 nM T52450 C2UAM8 10278729 IC50 = 116 nM T52450 C6KR5M 10278934 IC50 = 346.74 nM T52450 C3IG0K 10280852 IC50 = 6000 nM T52450 C80WUO 10282084 IC50 = 50000 nM T52450 C7TWG0 10289551 Ki > 4950 nM T52450 CJ63ER 10289607 Ki > 4950 nM T52450 CP0I5Y 10291146 IC50 > 10000 nM T52450 CJTV12 10293283 IC50 > 100000 nM T52450 CLP72J 10293348 IC50 > 10000 nM T52450 CS69YG 10293394 IC50 > 10000 nM T52450 CB82ZF 10294766 IC50 = 574 nM T52450 C89YGA 10295733 Ki > 2128 nM T52450 CDU36Y 10296475 Ki = 580 nM T52450 CTL3Y8 10296608 Ki > 4948 nM T52450 C48IRP 10296785 Ki = 210 nM T52450 CQ1Z0G 10298111 IC50 > 10000 nM T52450 CN14MI 10298369 Ki > 4949 nM T52450 CU5E9Z 10299198 Ki > 4948 nM T52450 C25EKM 10299665 Ki > 4900 nM T52450 CQ5BE8 10299709 IC50 = 78 nM T52450 C1BR6A 10300063 Ki > 4949 nM T52450 C80VEU 10300077 Ki > 4949 nM T52450 C8U3KW 10301524 IC50 > 50000 nM T52450 CFAU84 10301584 Ki > 4949 nM T52450 CP5AU1 10302088 Ki > 4949 nM T52450 C63BRA 10303333 IC50 > 50000 nM T52450 C4R9ZK 10311997 Ki > 4950 nM T52450 CE6MB0 10312141 Ki > 4350 nM T52450 C37ZDM 10317565 Ki = 3350 nM T52450 C59EDA 10317655 IC50 = 16 nM T52450 C2U6MY 10318916 Ki = 26 nM T52450 CNS0E8 10319540 IC50 = 230 nM T52450 CF4KT9 10320002 Ki > 4948 nM T52450 CG23FV 10320328 IC50 = 920 nM T52450 CC35NB 10321078 IC50 = 1560 nM T52450 CK4OG2 10321079 IC50 = 140 nM T52450 CJ6XM1 10321516 IC50 = 1012 nM T52450 CFQ4U0 10322451 Ki = 920 nM T52450 CY08WJ 10322755 Ki > 5000 nM T52450 C9DR2I 10323789 IC50 = 139 nM T52450 CQH5D4 10324032 IC50 = 54 nM T52450 CPI8R0 10324532 Ki = 2900 nM T52450 CSFZ76 10325592 Ki > 4949 nM T52450 CSG12E 10325620 IC50 = 12 nM T52450 C1C4VZ 10326004 Ki = 47800 nM T52450 CF5UN8 10326272 IC50 = 36 nM T52450 CP5Z4H 10326273 IC50 = 36 nM T52450 C5F0RK 10326931 IC50 = 190 nM T52450 CR6NX3 10340000 IC50 = 12 nM T52450 C7UZA4 10340758 IC50 = 89 nM T52450 CTC1E9 10341651 IC50 > 10000 nM T52450 CCK1A4 10342176 IC50 = 2100000 nM T52450 CFO74N 10343375 Ki = 2300 nM T52450 C7GK0A 10343478 IC50 = 17000 nM T52450 CJIW74 10343996 IC50 = 26 nM T52450 CW1VL2 10345348 IC50 = 1170 nM T52450 CPJ1G8 10345717 IC50 = 86 nM T52450 CX8H3Z 10346437 IC50 = 160 nM T52450 C94ANQ 10347529 IC50 = 284 nM T52450 CNP78B 10348836 Ki = 2200 nM T52450 C50DNH 10362338 Ki = 31 nM T52450 C9FU5G 10362663 IC50 = 320 nM T52450 CL4B2U 10364155 IC50 > 10000 nM T52450 CIJ5N7 10364252 IC50 = 25 nM T52450 CBA5I4 10365560 Ki = 5 nM T52450 CH89GT 10365752 IC50 = 10 nM T52450 C6WZ4F 10367355 IC50 = 88 nM T52450 C6FJU3 10367981 IC50 = 370 nM T52450 C8DJX4 10368307 Ki = 248 nM T52450 CT81YN 10370089 IC50 > 10 nM T52450 CJ96GA 10370197 IC50 = 56 nM T52450 CBTO07 10370226 Ki > 4949 nM T52450 C5VHS0 10370227 IC50 = 488 nM T52450 C6T4WO 10370281 Ki = 1068 nM T52450 CUA47P 10371161 Ki = 110 nM T52450 CP4BK2 10385954 IC50 = 740 nM T52450 C69LPF 10386446 IC50 = 760 nM T52450 C0IUQ7 10387351 Ki > 4948 nM T52450 C6G4PB 10387648 IC50 = 3.1 nM T52450 CEM0U7 10387692 IC50 = 490 nM T52450 CTQV87 10387878 IC50 = 55 nM T52450 C65AGQ 10388162 IC50 = 12 nM T52450 CS70LJ 10388253 IC50 > 10000 nM T52450 CL97HT 10388523 Ki > 850 nM T52450 C2Z8AO 10388678 IC50 = 470 nM T52450 C8CN6L 10388679 IC50 = 15600 nM T52450 CZNT94 10389113 IC50 2000 nM T52450 CP9WG5 10389610 IC50 = 322 nM T52450 CA2CL5 10389631 Ki = 3 nM T52450 CB6IH4 10389682 Ki = 350 nM T52450 CE5LQ8 10389828 IC50 = 44 nM T52450 CFN85O 10389832 IC50 = 10 nM T52450 CY2G0R 10391428 Ki > 4949 nM T52450 C8O1XU 10392082 IC50 = 6 nM T52450 CR38WZ 10392467 IC50 = 49 nM T52450 C8UTS7 10393307 IC50 = 22 nM T52450 C16BSA 10394828 IC50 = 30000 nM T52450 CFKA79 10395015 Ki > 2000 nM T52450 C9HM1A 10402302 IC50 > 10000000 nM T52450 CLP05D 10407603 IC50 = 1.2 nM T52450 CTX2S3 10410319 Ki = 167 nM T52450 CRD6Z4 10410935 IC50 = 86 nM T52450 CZ90OC 10412486 Ki = 2 nM T52450 C7V9JZ 10412739 IC50 = 1360 nM T52450 CA0TY8 10413076 Ki = 496 nM T52450 C98HMP 10413940 Ki = 1448 nM T52450 CJ95UZ 10414150 IC50 = 37 nM T52450 C7K0HG 10414437 Ki > 5000 nM T52450 CSY73P 10414917 IC50 = 44.67 nM T52450 CH1S2G 10414974 Ki = 1700 nM T52450 CV4JT6 10415842 IC50 = 70 nM T52450 C4J7IP 10416507 Ki = 720 nM T52450 CZ3D4T 10428502 IC50 = 15 nM T52450 C31TIX 10428779 IC50 = 40 nM T52450 CBL61N 10430546 IC50 = 150 nM T52450 CMO4U6 10431654 IC50 = 23 nM T52450 CCD1B8 10433014 IC50 = 1400 nM T52450 C3MSK7 10433015 IC50 = 810 nM T52450 C1SJ4K 10435554 IC50 = 500 nM T52450 CT7GC3 10435637 IC50 = 1820 nM T52450 CS32HR 10435935 IC50 = 5 nM T52450 C67UJP 10436058 IC50 = 34 nM T52450 CO6VM2 10436776 IC50 = 81 nM T52450 C9QS8N 10438212 IC50 = 15 nM T52450 C5WV1N 10439082 Ki > 2000 nM T52450 CIW2G8 10453253 IC50 = 2 nM T52450 CA75GC 10453674 IC50 > 10000 nM T52450 C54UDR 10453826 IC50 = 6 nM T52450 CP9WB1 10454818 Ki = 5100 nM T52450 C6T8VC 10456675 Ki = 3 nM T52450 CG47BR 10457660 IC50 = 19 nM T52450 CA5W6I 10458439 IC50 = 54 nM T52450 CP13CG 10459563 IC50 = 84 nM T52450 CA7DM9 10474389 IC50 = 100 nM T52450 C48ETI 10476560 IC50 = 490 nM T52450 CWV9Q2 10477531 Ki = 6 nM T52450 CP30UC 10478059 Ki = 1600 nM T52450 C87WDS 10478481 Ki = 2270 nM T52450 CHG02V 10478612 Ki = 6.57 nM T52450 CTL4W3 10479018 IC50 = 50 nM T52450 C9VIP5 10479752 Ki = 9600 nM T52450 CI7U4Z 10481280 Ki = 5 nM T52450 CHL30D 10482442 IC50 = 108 nM T52450 CNQZ36 10483139 Ki > 10000 nM T52450 COT6G1 10492779 Ki > 200000 nM T52450 C9XC8Y 10493383 IC50 = 150 nM T52450 CO92UA 10494668 Ki > 200000 nM T52450 C9KHT4 10495552 Ki = 4170 nM T52450 CV8U1L 10497756 IC50 = 33300 nM T52450 CA7HT2 10498521 Ki = 21 nM T52450 C6KD0A 10498747 IC50 = 0.4 nM T52450 CL8O6I 10500340 Ki > 200 nM T52450 CGK80V 10500816 Ki > 100 nM T52450 CVID65 10500886 Ki = 28 nM T52450 CP37WK 10501527 Ki = 24 nM T52450 CK6YN5 10501862 Ki = 31 nM T52450 CK4E0P 10501888 Ki = 15000 nM T52450 CZ2UY0 10502046 IC50 = 18 nM T52450 C36OMW 10502172 IC50 = 560 nM T52450 C1EAW7 10502187 Ki > 200000 nM T52450 C9QE1B 10502327 Ki = 62 nM T52450 C5V8HJ 10502382 IC50 = 3 nM T52450 CJZ5T8 10502487 IC50 > 10000 nM T52450 CSN17G 10502708 IC50 = 1200 nM T52450 CZ1R5Q 10502869 Ki = 2500 nM T52450 CBNM82 10503128 IC50 = 5.7 nM T52450 CO9S5H 10503708 Ki = 12 nM T52450 C9LJR5 10503737 IC50 = 236 nM T52450 C5Y4IA 10504081 IC50 = 13700 nM T52450 C2C7TE 10504472 IC50 = 780 nM T52450 CT2NM3 10505241 Ki = 29 nM T52450 CV19QD 10505495 Ki = 6000 nM T52450 CH6S8Y 10505729 IC50 > 10000 nM T52450 C6D7JF 10506147 IC50 = 56000 nM T52450 C7S0DB 10506158 IC50 = 3660 nM T52450 C03MRW 10507152 Ki = 60 nM T52450 CC6H8T 10507755 Ki = 50 nM T52450 C9C5EL 10521197 IC50 = 5.4 nM T52450 CBT12Q 10522080 IC50 = 329 nM T52450 CC2F5Y 10522311 IC50 = 73 nM T52450 CXD8I5 10523292 Ki > 200 nM T52450 CZ36JW 10523383 IC50 = 29000 nM T52450 C90HBF 10523728 Ki = 32 nM T52450 CQEH42 10524134 IC50 = 20 nM T52450 CYU87N 10524260 IC50 = 109 nM T52450 COT07L 10525329 IC50 = 324 nM T52450 C61GSD 10525562 IC50 = 25 nM T52450 CYB53K 10525912 Ki = 62 nM T52450 C56YKL 10525916 IC50 = 47 nM T52450 C14XUW 10526101 IC50 = 81 nM T52450 CJK6G1 10526509 IC50 = 75 nM T52450 CWLD37 10526788 IC50 = 300 nM T52450 CHS9Q5 10527785 IC50 = 450 nM T52450 CJ0D7G 10528505 IC50 = 54 nM T52450 CYGU41 10529315 IC50 > 10000 nM T52450 CGK37L 10529602 IC50 = 61.66 nM T52450 CQ82VY 10530944 Ki = 94 nM T52450 C86EWV 10541018 IC50 > 100000 nM T52450 CGE54K 10543918 Ki = 41000 nM T52450 CB7TX1 10543975 Ki > 200000 nM T52450 CO2R0P 10544323 IC50 = 1260 nM T52450 CQJA07 10544993 Ki = 17000 nM T52450 C0WHA9 10546565 Ki = 30 nM T52450 C40ZXE 10547784 Ki = 24 nM T52450 C4PK0U 10549114 IC50 = 3 nM T52450 C4TA1K 10549256 IC50 = 3 nM T52450 C5JS8L 10549329 IC50 = 43.65 nM T52450 CHCI01 10549577 IC50 = 210 nM T52450 CG27UI 10549756 Ki = 87 nM T52450 C2HJ1U 10549764 IC50 = 227 nM T52450 C82HQE 10550145 Ki = 54 nM T52450 CRHP20 10550304 IC50 = 219 nM T52450 C7WQ5Z 10550399 IC50 = 110 nM T52450 CNQ75F 10551139 IC50 = 1059 nM T52450 CCH0K3 10551483 IC50 = 92 nM T52450 CC2FM6 10551489 IC50 > 10000 nM T52450 C5UD0A 10551910 IC50 = 56000 nM T52450 CNE73L 10552476 IC50 = 325 nM T52450 CU8QP7 10552732 Ki = 17 nM T52450 CI8XG0 10554869 IC50 = 41000 nM T52450 CZ41HP 10554978 Ki > 100 nM T52450 CD3R8V 10562830 IC50 = 3136.72 nM T52450 CT7O9M 10569678 IC50 = 2200 nM T52450 C8RWE4 10569743 IC50 = 26000 nM T52450 CE14GM 10570702 IC50 = 1500 nM T52450 C2MD1V 10571436 IC50 = 7120 nM T52450 CBXZ79 10572150 IC50 = 220 nM T52450 CPF0R5 10572544 Ki = 5000 nM T52450 CYX52N 10572651 Ki = 32000 nM T52450 C21VZS 10573362 IC50 = 90 nM T52450 CS9Y3Q 10573446 IC50 = 19 nM T52450 C42IAF 10573603 Ki = 59 nM T52450 CG39CF 10574279 Ki = 33 nM T52450 C61IUN 10574937 IC50 = 1.9 nM T52450 C9YFC5 10577526 IC50 = 36 nM T52450 C1KH7E 10578728 IC50 > 10000 nM T52450 CM4XT6 10578789 IC50 = 102 nM T52450 CK05ZH 10579086 Ki = 55 nM T52450 C9L5OM 10579282 IC50 = 79 nM T52450 C8J6HS 10591505 Ki > 200 nM T52450 CIUO27 10593253 IC50 = 155 nM T52450 CB20LM 10594000 Ki = 60 nM T52450 CUTS47 10594564 IC50 = 18000 nM T52450 CN4Y6H 10594565 IC50 = 14000 nM T52450 CUN73L 10595134 Ki = 52000 nM T52450 CI71CK 10595804 Ki = 18 nM T52450 CYNC76 10596158 IC50 = 13000 nM T52450 CD65NF 10597516 Ki = 36 nM T52450 CP2H8O 10597673 Ki = 15 nM T52450 C0R8ND 10599533 IC50 = 19 nM T52450 CQCW86 10599579 IC50 = 26 nM T52450 CW18QK 10599594 IC50 = 19 nM T52450 CR1JI4 10600645 IC50 > 1000 nM T52450 CL4UB6 10600908 IC50 = 1.5 nM T52450 C6RH4O 10601640 IC50 = 87 nM T52450 C02RNF 10602071 IC50 = 1.1 nM T52450 CZ7QK1 10602072 IC50 = 1.2 nM T52450 CEJ1U0 10603377 Ki > 100 nM T52450 C5G9MI 10610114 Ki = 900 nM T52450 C84URB 10610500 Ki > 100000 nM T52450 CG32FM 10613145 IC50 = 300 nM T52450 CZD9B3 10617580 IC50 = 64 nM T52450 CL02BO 10618584 IC50 = 3200 nM T52450 C06CAN 10619639 Ki = 24 nM T52450 CV14UH 10619971 Ki = 19 nM T52450 CM06XN 10620633 IC50 = 6790 nM T52450 C8IZN2 10620836 IC50 = 35 nM T52450 CW1DA5 10621015 IC50 = 2.2 nM T52450 C0JGS3 10621776 IC50 = 500 nM T52450 CL5QN9 10622296 IC50 = 68 nM T52450 CL62YC 10622822 IC50 = 0.5 nM T52450 CZJB31 10622970 IC50 = 158 nM T52450 CL67UQ 10623250 IC50 > 10000 nM T52450 CQH75Y 10624313 Ki = 6200 nM T52450 CXV87K 10625636 IC50 = 20.89 nM T52450 CGB29T 10625771 IC50 = 260 nM T52450 C98KGO 10625860 IC50 = 49 nM T52450 C70MFZ 10626445 Ki > 100 nM T52450 C5VGB1 10626732 Ki > 100 nM T52450 CL43CO 10627365 IC50 = 2322 nM T52450 C8UY9P 10639050 IC50 > 30000 nM T52450 CA63VQ 10640307 Ki = 26 nM T52450 CPFH58 10641536 IC50 > 40000 nM T52450 C7KGM3 10642071 IC50 = 22 nM T52450 CWRY91 10642128 IC50 = 115 nM T52450 CI2QB9 10642965 IC50 = 13 nM T52450 C41RKE 10643401 Ki = 25 nM T52450 CUAI71 10643973 Ki = 37 nM T52450 C2O1XM 10647817 IC50 = 80 nM T52450 CVX7Q2 10648390 Ki = 26 nM T52450 CNF9I2 10648570 IC50 = 25 nM T52450 C5RWF4 10648802 IC50 = 31 nM T52450 CX48UV 10649092 IC50 = 700 nM T52450 C6S1KA 10649216 IC50 > 10000 nM T52450 CM4JF2 10649665 IC50 = 2.6 nM T52450 COT6B8 10650624 Ki > 100 nM T52450 C69SPO 10650906 Ki = 54 nM T52450 CT23XW 10650907 Ki = 49 nM T52450 C27QHB 10663143 IC50 = 175 nM T52450 CGSX70 10664302 IC50 = 120 nM T52450 C97KZU 10665624 IC50 = 4200 nM T52450 CF0E6H 10668745 IC50 = 4200 nM T52450 C4HJS1 10669027 Ki = 2000 nM T52450 CFYC35 10669215 Ki = 41 nM T52450 C6TC0Z 10669216 Ki = 34 nM T52450 C8HK0C 10669534 IC50 = 81 nM T52450 CAI72H 10670246 IC50 = 1200 nM T52450 CY6QC1 10670819 IC50 = 354 nM T52450 C4QVL0 10670896 Ki = 46 nM T52450 CPG5O2 10671155 IC50 = 99 nM T52450 CWB19K 10671441 Ki = 6 nM T52450 C09LJR 10671827 IC50 = 68 nM T52450 C17LYV 10672346 IC50 > 10000 nM T52450 CMU74I 10672857 IC50 > 10000 nM T52450 CBO26H 10687032 IC50 = 638 nM T52450 CXTP56 10688727 IC50 = 10 nM T52450 C0OJ9C 10689683 IC50 = 150 nM T52450 CSA80H 10692194 IC50 = 310 nM T52450 CS5CL7 10692307 IC50 = 39 nM T52450 CR5KF8 10692994 IC50 = 100000 nM T52450 CDI12G 10693559 IC50 = 0.7 nM T52450 CB70DA 10693592 IC50 = 2000 nM T52450 C8JX1G 10693698 Ki = 43 nM T52450 CVML68 10693881 IC50 = 87 nM T52450 CWS4N1 10695749 IC50 = 1.7 nM T52450 CZGC63 10695865 IC50 = 11500 nM T52450 CVQF97 10695971 IC50 = 140 nM T52450 CW6CF7 10696226 IC50 = 74 nM T52450 C6MWX8 10696713 IC50 = 1320 nM T52450 C1YFC3 10696977 IC50 > 10000 nM T52450 C4BME8 10697140 IC50 > 10000 nM T52450 CG5JM9 10698412 Ki = 58 nM T52450 C56VSE 10698786 Ki = 50 nM T52450 C5E8QF 10707457 Ki > 200 nM T52450 C7CI4T 10713194 Ki = 8900 nM T52450 CJZ0X3 10714009 Ki = 16000 nM T52450 CG38ZD 10714323 IC50 = 3100 nM T52450 C2GL3A 10714610 Ki = 2000 nM T52450 C4IWF2 10714988 IC50 = 280 nM T52450 CO9KV7 10715115 IC50 = 26 nM T52450 CE1D6G 10716217 IC50 < 1 nM T52450 CF98LK 10716463 Ki = 12000 nM T52450 CF51EI 10716486 IC50 = 62 nM T52450 C0ZX6T 10717308 IC50 = 7000 nM T52450 C3TGW8 10717400 Ki > 200 nM T52450 CQZ7M8 10718133 Ki = 25 nM T52450 C7OSW8 10718200 IC50 = 17 nM T52450 CI64YZ 10718883 IC50 = 70 nM T52450 CVPC97 10718960 IC50 = 23.99 nM T52450 C35MRE 10719092 IC50 = 32 nM T52450 CVW81M 10719595 IC50 > 10000 nM T52450 C4RD0P 10719602 Ki = 29000 nM T52450 CF46SQ 10721337 Ki > 100 nM T52450 C4J1WN 10721454 IC50 = 240 nM T52450 CC1FB8 10721904 Ki = 53 nM T52450 CB2QD0 10723468 Ki = 79 nM T52450 CG4DA0 10731747 IC50 = 2510 nM T52450 C0TI1M 10734897 IC50 = 1290 nM T52450 C8KE2C 10735676 IC50 = 65 nM T52450 CBHX39 10736792 Ki = 21000 nM T52450 CO7VP4 10737552 Ki = 21 nM T52450 C51DZG 10737732 IC50 = 6500 nM T52450 C1LS5U 10738104 IC50 = 170 nM T52450 CL74TG 10738165 IC50 = 15 nM T52450 C76ANK 10739335 IC50 = 8 nM T52450 CB8G2D 10739728 Ki = 22 nM T52450 C0T2VK 10740460 IC50 = 115 nM T52450 C4FWC9 10740485 Ki > 200 nM T52450 CKJD45 10741133 IC50 = 24000 nM T52450 C0WKL7 10741470 Ki = 9 nM T52450 CL64BU 10741592 IC50 = 2.3 nM T52450 C0QT2F 10741956 Ki = 31 nM T52450 C4MQ8L 10742072 IC50 = 100 nM T52450 CKX5R3 10742142 IC50 = 3340 nM T52450 CHW23E 10742387 IC50 = 1.2 nM T52450 CY2BZ0 10742536 Ki = 83 nM T52450 CCH94Q 10743507 IC50 = 60 nM T52450 CTA0Y4 10743933 IC50 = 37 nM T52450 C5BZ0J 10745489 Ki = 89 nM T52450 C9ILP3 10745718 IC50 = 40000 nM T52450 CK30AE 10745748 Ki = 72 nM T52450 CWF50D 10745851 Ki = 95 nM T52450 CMZC64 10756622 IC50 = 297 nM T52450 CE09PI 10757715 IC50 = 250 nM T52450 CA3F1N 10758013 IC50 = 144.54 nM T52450 CTKR07 10758266 Ki > 200000 nM T52450 CLEG16 10761206 Ki = 2160 nM T52450 CDX13Z 10761730 Ki = 14 nM T52450 CA4U7D 10762262 Ki = 24 nM T52450 C68THN 10763851 IC50 = 81 nM T52450 CM54WS 10764477 Ki = 900 nM T52450 CAG53Y 10764489 IC50 = 42 nM T52450 C0ZJB9 10764600 IC50 = 994 nM T52450 CJE76M 10764871 IC50 = 2000 nM T52450 CQ0KM4 10765140 IC50 = 19 nM T52450 COAL70 10765803 IC50 = 310 nM T52450 C3P2TS 10766036 IC50 = 24800 nM T52450 CA6C0Z 10766622 Ki = 6 nM T52450 CN6P1J 10766950 IC50 = 270 nM T52450 CWR5Z3 10767105 IC50 > 10000 nM T52450 CR4I1E 10767157 IC50 > 10000 nM T52450 C7Q2EM 10767236 IC50 = 350 nM T52450 C1M8BZ 10767542 IC50 > 1000 nM T52450 CN83AJ 10768085 IC50 = 40.74 nM T52450 CQ7J4I 10769007 IC50 > 10000 nM T52450 CQ6U2Y 10780743 Ki = 75 nM T52450 CIN4A9 10783989 Ki = 1000 nM T52450 C31KWI 10785840 Ki = 20000 nM T52450 C15PVT 10785952 Ki = 30 nM T52450 CLAP90 10785969 IC50 > 1000 nM T52450 C2FA7J 10787997 IC50 = 140 nM T52450 C16XQR 10788211 IC50 = 42 nM T52450 C0DFB9 10788617 IC50 = 1 nM T52450 CNAE08 10788733 IC50 = 3600 nM T52450 CXQD12 10789326 IC50 > 10000 nM T52450 CKV2O8 10789493 IC50 = 22 nM T52450 CM74LH 10789594 IC50 > 1000 nM T52450 C45UGJ 10789671 IC50 = 20 nM T52450 C9NZ4W 10789711 IC50 = 18 nM T52450 CHWG02 10790787 IC50 = 6510 nM T52450 CF4T1N 10791150 Ki = 1800 nM T52450 C3P7LZ 10792025 IC50 = 15.85 nM T52450 CWCD73 10805054 IC50 = 90 nM T52450 C1WZ4S 10805349 IC50 = 49.5 nM T52450 C9VML0 10807861 Ki = 226000 nM T52450 C6FWC1 10808125 IC50 = 2.9 nM T52450 CN8I3Z 10808172 IC50 = 1548 nM T52450 CQX5P6 10808260 IC50 = 380 nM T52450 C5HF8Z 10809178 IC50 = 64 nM T52450 CT1AI4 10810573 IC50 = 260 nM T52450 CU9F7V 10810684 IC50 = 53.7 nM T52450 CV3ZA5 10812444 IC50 = 228 nM T52450 CZB7L2 10812929 IC50 = 2.9 nM T52450 C4TF0K 10813874 IC50 = 127 nM T52450 CCIL63 10813879 IC50 = 230 nM T52450 CIUN51 10814028 IC50 > 10000 nM T52450 C80CZA 10815208 IC50 = 827 nM T52450 C34KQG 10816626 IC50 = 72.44 nM T52450 CS7BY4 10816934 IC50 = 15000 nM T52450 CBL54W 10816989 IC50 = 107.15 nM T52450 CX2E1C 10829071 IC50 = 23 nM T52450 C3AI5Z 10831752 IC50 = 8600 nM T52450 CLK9P7 10832592 IC50 = 688 nM T52450 CF50HD 10832925 IC50 = 50000 nM T52450 COE82D 10833334 IC50 = 154.88 nM T52450 C5OG4U 10833497 IC50 = 12000 nM T52450 C2A0IX 10833840 IC50 = 92 nM T52450 CH90ZB 10834348 IC50 = 13 nM T52450 C9M1JI 10834357 IC50 = 42.66 nM T52450 C48PYQ 10836923 IC50 = 30 nM T52450 CH8OV4 10837276 IC50 = 271 nM T52450 CF40VH 10837557 IC50 = 270 nM T52450 CR0E9Q 10837740 Ki = 30 nM T52450 CY4J9A 10838149 IC50 = 440 nM T52450 CR50UM 10839419 Ki = 25 nM T52450 CA76MU 10840059 IC50 > 10000 nM T52450 C6SDH4 10840060 IC50 = 2.4 nM T52450 CL1KG7 10840630 Ki > 100 nM T52450 CEG8T6 10852576 IC50 = 518 nM T52450 CN5MJ6 10853865 IC50 > 30000 nM T52450 C3UCL2 10854279 IC50 = 70 nM T52450 C0W6AK 10854448 Ki > 200000 nM T52450 C9EU2B 10854874 Ki = 67000 nM T52450 C6ZSP8 10862104 Ki > 4949 nM T52450 CQ1L7C 10863755 Ki > 4949 nM T52450 CF72UK 10864417 IC50 = 18 nM T52450 C6CD3R 10873386 Ki < 1 nM T52450 C0AQL8 10873958 Ki > 4949 nM T52450 CBQ70P 10874312 IC50 = 126 nM T52450 CLG40T 10874819 IC50 = 50000 nM T52450 CXY47P 10875332 IC50 > 100000 nM T52450 CXGN38 10875470 IC50 > 2500 nM T52450 CJ0LE4 10876254 Ki > 2000 nM T52450 CIB8Y1 10884337 Ki > 4949 nM T52450 C3AY8O 10885569 IC50 > 1000 nM T52450 CAU0I3 10885834 IC50 = 1850 nM T52450 CG1I4Y 10886343 IC50 = 2180 nM T52450 CF5L1R 10886549 IC50 = 593 nM T52450 CA64PN 10886607 IC50 = 76 nM T52450 CDZ04P 10887027 Ki > 2000 nM T52450 C0R5QL 10894433 Ki = 4.59 nM T52450 C7AMS4 10895808 Ki > 4949 nM T52450 CPJ0I8 10896934 IC50 = 5400 nM T52450 CU7YE0 10896986 IC50 = 5.1 nM T52450 CMV89R 10897017 IC50 = 57 nM T52450 C3FQT7 10903871 Ki = 2288 nM T52450 CX93MR 10907320 IC50 > 10000 nM T52450 CM9G8A 10907701 IC50 = 50000 nM T52450 CSK87I 10907725 IC50 = 21 nM T52450 C13CJH 10907740 IC50 > 50000 nM T52450 C69ZTR 10913644 Ki > 4949 nM T52450 C2QR0W 10914151 Ki = 4000 nM T52450 CAH70N 10914350 IC50 = 49 nM T52450 C2M4PK 10916140 Ki = 759 nM T52450 C7XE3L 10917417 Ki = 2019 nM T52450 CGI2T1 10928606 IC50 > 36000 nM T52450 CXHA75 10928874 IC50 = 2760 nM T52450 C40PRC 10929100 IC50 = 423 nM T52450 CXY4L6 10929354 IC50 > 1000 nM T52450 CDSQ41 10929404 IC50 > 70000 nM T52450 CLIR35 10938505 IC50 = 1260 nM T52450 C1QVT6 10939850 IC50 = 990 nM T52450 CWO29J 10940364 IC50 = 2100 nM T52450 CL64UM 10940712 IC50 = 8.1 nM T52450 C89IYC 10948209 Ki = 143 nM T52450 C7GH8P 10948665 Ki < 1 nM T52450 C2TA9N 10949166 Ki = 4.58 nM T52450 CC46WL 10950008 Ki > 5000 nM T52450 C9YOU4 10951375 IC50 = 164 nM T52450 CJI1G0 10951750 IC50 = 16 nM T52450 C0A2IR 10958121 Ki = 335 nM T52450 C3K1BL 10959017 IC50 = 100 nM T52450 C7PX8G 10960109 Ki > 850 nM T52450 C5HS4F 10961382 Ki > 4949 nM T52450 CMY8S6 10961569 IC50 = 5200 nM T52450 CPA1Q2 10961828 IC50 > 50000 nM T52450 C5ZV9Q 10962137 IC50 = 51 nM T52450 C30FBA 10970628 Ki > 5000 nM T52450 CQ68IE 10972732 IC50 = 3.6 nM T52450 CJHO94 10972891 IC50 > 50000 nM T52450 CTP6I0 10973485 IC50 = 6700 nM T52450 C9DM0P 10980832 Ki = 497 nM T52450 CL7K8S 10983560 Ki < 1 nM T52450 C3UH2B 10983665 Ki > 4949 nM T52450 CR9J5B 10983887 IC50 > 10000 nM T52450 C68LPK 10983913 IC50 = 2500 nM T52450 CJ8I9G 10983916 IC50 = 38 nM T52450 CS7D0Z 10984030 IC50 = 280 nM T52450 C0NIX9 10985227 IC50 > 2700 nM T52450 CSI5G1 10992109 IC50 = 10 nM T52450 C0G8TE 10993343 Ki > 5000 nM T52450 CW8Z6R 10993677 Ki > 4949 nM T52450 CCX0L6 10994350 IC50 = 188 nM T52450 CW0Y6I 10994897 IC50 = 240 nM T52450 CA5I7L 10995373 IC50 = 85 nM T52450 C3QX0T 11005761 IC50 = 44 nM T52450 CJM41O 11006091 IC50 = 820 nM T52450 C4PNK3 11006191 IC50 = 19610 nM T52450 C95NXQ 11006894 Ki > 2000 nM T52450 C7WEZ4 11009332 Ki = 40000 nM T52450 CS4FL3 11012667 IC50 = 300 nM T52450 C5JE9G 11014504 IC50 = 583 nM T52450 C8ERT5 11014626 Ki > 850 nM T52450 C75DGS 11015731 Ki = 35.6 nM T52450 CBE68H 11016073 Ki = 550 nM T52450 CG2DK0 11016448 IC50 = 1400 nM T52450 C3IYK8 11016511 IC50 = 90 nM T52450 CF30UR 11016519 IC50 = 297 nM T52450 CODQ51 11016616 IC50 = 1370 nM T52450 CO6C8A 11017232 IC50 = 188 nM T52450 CM1H5P 11026185 Ki = 5.3 nM T52450 CQD70Y 11026301 Ki = 125 nM T52450 C6IHF5 11026991 IC50 > 100000 nM T52450 C3LF1Y 11027584 Ki > 4949 nM T52450 CF5KU1 11027718 IC50 > 50000 nM T52450 CA49QF 11027968 IC50 = 9900 nM T52450 CLXZ15 11037377 Ki = 10.7 nM T52450 C0ERN9 11037836 Ki = 6.23 nM T52450 CT2S0G 11038175 IC50 > 50000 nM T52450 C83AKP 11038896 IC50 = 100 nM T52450 CG3B5N 11039339 IC50 = 110 nM T52450 C3W9IT 11046880 Ki = 946 nM T52450 CZO40T 11048604 Ki = 573 nM T52450 C5R7JX 11049650 Ki > 4949 nM T52450 CW42KO 11049937 IC50 = 8000 nM T52450 CQ08SN 11049982 IC50 > 50000 nM T52450 CYA27S 11059553 Ki < 1 nM T52450 C9RU4I 11059620 IC50 = 5210 nM T52450 CH8O1E 11060081 Ki > 4949 nM T52450 CM6X1E 11061555 Ki > 2000 nM T52450 C49PNL 11069047 Ki = 1.4 nM T52450 C1N5PT 11070986 IC50 = 4900 nM T52450 C18EIZ 11071831 IC50 = 1220 nM T52450 C2LSU0 11072397 IC50 = 96 nM T52450 CM9EP0 11077031 IC50 = 647 nM T52450 C5MUD2 11078779 IC50 = 78 nM T52450 C43JOG 11080156 Ki > 5000 nM T52450 C7VKE3 11080910 Ki < 1 nM T52450 CT3VX4 11080936 Ki > 4949 nM T52450 CG0A4C 11081333 IC50 = 10000 nM T52450 CVJX34 11081788 Ki < 1 nM T52450 C05MUK 11081992 IC50 = 1450 nM T52450 C6XI8J 11082293 IC50 = 26 nM T52450 CUNM68 11083152 Ki > 4949 nM T52450 CF0NJ9 11090097 IC50 = 5 nM T52450 CS29GX 11091928 IC50 > 100000 nM T52450 C16WBE 11092175 IC50 = 540 nM T52450 CE8V9B 11092295 IC50 = 396 nM T52450 CR8ZA7 11092551 IC50 = 63000 nM T52450 CT2CH7 11092701 IC50 > 50000 nM T52450 C6R7XB 11092861 Ki > 4949 nM T52450 CWT6C7 11092884 IC50 = 108 nM T52450 CX69YN 11093502 IC50 = 49 nM T52450 C8CK3E 11102531 IC50 = 93 nM T52450 C57OXT 11102540 Ki = 2.21 nM T52450 CA2OS3 11103408 IC50 = 24 nM T52450 C6G2DI 11111616 Ki > 4949 nM T52450 CUK03P 11112062 Ki = 4747 nM T52450 CWV45Z 11112302 Ki > 4949 nM T52450 CEAI92 11112993 IC50 = 40 nM T52450 CY1SR9 11113744 IC50 > 10000 nM T52450 CI1GS5 11114351 IC50 = 144 nM T52450 CUO7B3 11122933 Ki = 1.8 nM T52450 CNGP50 11122963 IC50 = 4500 nM T52450 CB2I5K 11123701 IC50 = 10 nM T52450 C8YVE5 11123989 IC50 > 10000 nM T52450 C3PR1J 11124862 IC50 = 122 nM T52450 CAJ27B 11124943 IC50 = 52 nM T52450 CNBG53 11124956 IC50 = 36 nM T52450 CX2B6C 11125147 Ki > 2000 nM T52450 C9GJ7C 11133809 Ki > 4949 nM T52450 C2YBQ7 11134935 IC50 = 3490 nM T52450 C8DMW5 11135133 IC50 > 100000 nM T52450 CD3N8B 11135304 IC50 = 532 nM T52450 CPO02F 11142863 IC50 = 1380 nM T52450 CF52TX 11143173 Ki = 30953 nM T52450 C3V4ZX 11143285 IC50 = 299 nM T52450 CH61QF 11144824 IC50 > 50000 nM T52450 C8HM2R 11145437 Ki > 4949 nM T52450 CHF19X 11146467 Ki > 4949 nM T52450 C5WS3E 11147931 IC50 = 50000 nM T52450 CVI3F8 11188429 IC50 > 10000 nM T52450 CCQ6N8 11194666 IC50 > 100000 nM T52450 CO5VN2 11201367 IC50 > 10000 nM T52450 CO76XI 11205873 IC50 = 50000 nM T52450 C9R7OM 11207122 IC50 = 70000 nM T52450 C72UCB 11233687 IC50 = 4567 nM T52450 CPV9L7 11246575 Ki = 128 nM T52450 CUOH67 11252195 IC50 > 100000 nM T52450 CJZ3P6 11257884 Ki > 5000 nM T52450 CD1FT8 11258906 IC50 = 96 nM T52450 CO7T3M 11261246 IC50 = 3000 nM T52450 CC62RY 11279665 IC50 = 257.04 nM T52450 CP17ID 11284983 IC50 = 30000 nM T52450 CF9O2R 11286824 IC50 = 40000 nM T52450 C1IW7N 11292680 IC50 = 147 nM T52450 C8C5AV 11294179 Ki > 4948 nM T52450 CK91YW 11317404 IC50 > 5000 nM T52450 CLH50U 11318841 IC50 = 23400 nM T52450 CJ5SU9 11328354 Ki > 300000 nM T52450 CN2P4G 11328571 IC50 > 5000 nM T52450 C0XR3B 11330861 IC50 = 37100 nM T52450 C49CDU 11335940 IC50 > 98000 nM T52450 CQH57S 11342435 IC50 > 400000 nM T52450 CZ8B0D 11349945 Ki = 318 nM T52450 CCKI02 11360440 Ki = 26 nM T52450 C7QNX8 11363138 IC50 > 5000 nM T52450 CM8Y1J 11367571 IC50 = 80000 nM T52450 CTQK48 11373358 Ki > 4949 nM T52450 C48DYJ 11374008 Ki > 850 nM T52450 CL8QO7 11382562 IC50 = 3000 nM T52450 CNZ0T5 11386918 IC50 = 3963 nM T52450 CUJ4V0 11391937 IC50 = 3301.33 nM T52450 C9KVB7 11394505 IC50 = 274 nM T52450 C13NCF 11400989 IC50 = 20000 nM T52450 C3EX5J 11407165 Ki = 162 nM T52450 C2EUO5 11417011 IC50 > 10000 nM T52450 CK95HW 11429232 Ki = 938 nM T52450 C01FLQ 11441438 Ki = 3166 nM T52450 CI0V6L 11447356 IC50 > 100000 nM T52450 C5NAJ3 11449819 IC50 = 1146 nM T52450 COS67B 11456566 IC50 = 60000 nM T52450 CCMT46 11457732 IC50 > 100000 nM T52450 CQ1D6E 11470070 IC50 = 30000 nM T52450 C1KP2Q 11473879 Ki > 4949 nM T52450 C5QEZ8 11483818 IC50 = 1509 nM T52450 CJ46KN 11508259 Ki = 160 nM T52450 CWS35C 11510523 IC50 > 50000 nM T52450 C5G8PM 11511807 IC50 > 5000 nM T52450 C5VUM2 11517085 Ki = 18700 nM T52450 C5MO0U 11526826 IC50 > 100000 nM T52450 C9Y6LH 11533683 IC50 > 50000 nM T52450 C2OA3K 11547967 IC50 > 5000 nM T52450 C1NZB9 11548265 IC50 = 700 nM T52450 CIWP38 11555036 IC50 = 753 nM T52450 CO9BC3 11562986 IC50 > 5000 nM T52450 CW5A4S 11569716 IC50 > 100000 nM T52450 CHV2G1 11575995 Ki > 10000000 nM T52450 C3H2DG 11577137 IC50 > 5000 nM T52450 CM6GO2 11577517 IC50 > 5000 nM T52450 C0Q5FU 11592023 IC50 > 5000 nM T52450 CSQ5M8 11598899 IC50 > 5000 nM T52450 CTQ87G 11599024 IC50 > 50000 nM T52450 CVGC49 11603611 Ki = 0.7 nM T52450 CUL5H2 11605631 IC50 = 259 nM T52450 C0VCJ8 11613810 IC50 > 100000 nM T52450 CXKU59 11620780 IC50 > 5000 nM T52450 CCBS59 11634234 IC50 = 8780 nM T52450 CNY92D 11640694 Ki > 90000 nM T52450 CFV49P 11641262 IC50 = 8660 nM T52450 CU6S3J 11655819 IC50 = 309.03 nM T52450 CK9F4P 11673778 IC50 > 2000 nM T52450 CFC74O 11678245 IC50 > 5000 nM T52450 CY0T4D 11685065 IC50 > 5000 nM T52450 CRF7V9 11691964 IC50 > 100000 nM T52450 CKGR97 11692294 IC50 > 5000 nM T52450 C3U6ZR 11697504 Ki > 50000 nM T52450 C6PM1J 11713686 IC50 > 5000 nM T52450 C1MJ3P 11713694 IC50 > 5000 nM T52450 C2BJ3X 11716217 Ki = 3300 nM T52450 C4ECU2 11720597 IC50 > 5000 nM T52450 CCD93H 11730086 Ki = 300 nM T52450 CBT48P 11731926 Ki = 7.8 nM T52450 CA43HK 11732287 Ki = 10.5 nM T52450 C68KBY 11732585 Ki > 4949 nM T52450 C7CED0 11733417 IC50 > 10000 nM T52450 CI0KL2 11733573 IC50 > 10000 nM T52450 C64LQC 11733862 Ki > 5000 nM T52450 C27SBC 11734162 IC50 = 490 nM T52450 CIU03K 11734219 Ki > 4949 nM T52450 C1Q9YR 11741600 IC50 = 30 nM T52450 CNW82E 11744630 IC50 = 150 nM T52450 CJOE40 11748355 Ki = 92 nM T52450 C4HD9K 11751106 IC50 > 5000 nM T52450 C6HV8Z 11752434 IC50 = 430 nM T52450 CO8QT0 11753905 Ki > 4948 nM T52450 C3N1WB 11754235 Ki = 140 nM T52450 C3P0TZ 11754739 Ki = 8400 nM T52450 CJ4G5D 11754907 IC50 = 301 nM T52450 CE6OS0 11755521 IC50 = 22 nM T52450 C5E7KU 11757592 Ki = 61 nM T52450 CUC9R5 11758082 IC50 = 19 nM T52450 CZ5V9G 11758096 IC50 = 29 nM T52450 CF2J8V 11758099 IC50 > 10000 nM T52450 C2KU3D 11760296 IC50 = 262 nM T52450 C3RW1X 11761191 Ki < 1 nM T52450 C6K8HR 11761578 Ki > 4949 nM T52450 CE1HZ4 11761760 Ki < 1 nM T52450 C04DFH 11783486 Ki = 3.5 nM T52450 C7BV5P 11792968 IC50 = 138.04 nM T52450 CKM6P2 11795228 IC50 = 996 nM T52450 CCSD72 11795621 IC50 = 1.9 nM T52450 CY8N1U 11795715 Ki = 39 nM T52450 CY7H2T 11795824 Ki = 18 nM T52450 CK24XT 11796481 Ki = 14 nM T52450 C46KHU 11796490 IC50 = 1.9 nM T52450 C47OIA 11797154 IC50 = 33 nM T52450 CHB01Z 11797196 IC50 = 74 nM T52450 CJ4VL3 11797382 IC50 > 1000 nM T52450 CKUM64 11797718 IC50 = 37 nM T52450 CCD4W2 11797992 IC50 = 493 nM T52450 CHQR96 11798386 IC50 = 24 nM T52450 CGL39X 11798547 Ki = 1500 nM T52450 C19RCP 11799753 Ki = 25 nM T52450 C2YD4N 11809525 IC50 = 211 nM T52450 C1NRV6 11811437 IC50 = 139 nM T52450 CQ9HE2 11811551 IC50 = 3890 nM T52450 CSG07A 11811629 Ki = 686 nM T52450 CK03NI 11811717 Ki > 5000 nM T52450 CLW3F1 11812791 IC50 = 6050 nM T52450 C20PYA 11813392 IC50 = 2000 nM T52450 CH3SV6 11813493 IC50 = 5900 nM T52450 CZ08ID 11814382 IC50 = 133 nM T52450 C8DY3Z 11817193 IC50 > 100000 nM T52450 CEN02U 11822212 Ki > 4949 nM T52450 CDU9S2 11824087 Ki = 732 nM T52450 C3VO5H 11824148 Ki = 0.6 nM T52450 C7BK5P 11825105 IC50 = 25 nM T52450 CKEM29 11827006 IC50 = 45000 nM T52450 CV2MX4 11832221 Ki = 221 nM T52450 C48QEH 11833533 Ki = 980 nM T52450 C02BWA 11967143 Ki > 2000 nM T52450 CB80OT 12000718 IC50 > 20000 nM T52450 C43PJZ 12000720 IC50 > 20000 nM T52450 CUQM03 12074753 IC50 = 770000 nM T52450 CKND02 12074756 IC50 = 1400000 nM T52450 C4I1TJ 12074757 IC50 > 10000000 nM T52450 CJ8W2C 12074758 IC50 > 10000000 nM T52450 C0JID3 12447203 Ki > 100000 nM T52450 CTHQ39 12635073 Ki = 33000 nM T52450 CIQX87 12635074 Ki = 74000 nM T52450 C0XKJ1 12671872 IC50 = 30000 nM T52450 CB1F2E 12971983 IC50 = 8020 nM T52450 CJY6X7 12971984 IC50 = 388 nM T52450 CZYE40 12971985 IC50 = 25900 nM T52450 CSR94V 13559594 IC50 = 5833.61 nM T52450 C71ASU 13644537 IC50 = 3246.57 nM T52450 C1AJO7 13968141 IC50 > 300000 nM T52450 CA2H8V 14303060 IC50 = 640 nM T52450 C5J1CE 14505615 Ki = 140000 nM T52450 C0XI2R 15296015 IC50 > 1000 nM T52450 C1IZ7D 15296597 IC50 = 57.54 nM T52450 CGH19T 15296844 IC50 > 300000 nM T52450 CKN3R1 15430588 IC50 = 361 nM T52450 C63MFQ 15435266 IC50 = 768 nM T52450 CH80JI 15435267 Ki = 7700 nM T52450 CZ0NL1 15484680 IC50 = 631 nM T52450 COZM90 15485452 IC50 = 10 nM T52450 CEM2O0 15485453 IC50 = 46 nM T52450 CT68FI 15487434 Ki > 10000 nM T52450 CJR3Z8 15487435 Ki > 10000 nM T52450 C46XNB 15487436 Ki > 10000 nM T52450 C16TEM 15516782 IC50 = 4000 nM T52450 CV1HA9 15516783 IC50 > 10000 nM T52450 CEKN36 15520981 IC50 = 59 nM T52450 CP2C4Z 15524387 Ki = 75000 nM T52450 CAF7R5 15524388 Ki = 1163 nM T52450 C17HGN 15524389 Ki = 95500 nM T52450 CFH8Y6 15524390 Ki = 50000 nM T52450 C47RXG 15541745 IC50 = 8000 nM T52450 CEFV16 15541746 IC50 = 6300 nM T52450 C1GW2T 15541747 IC50 = 5000 nM T52450 CU05VE 15541748 IC50 = 9000 nM T52450 CXUG10 15546245 IC50 = 900 nM T52450 CU7CM3 15551877 IC50 = 176 nM T52450 C5TLB4 15765753 IC50 = 5516.37 nM T52450 CO2XY0 15851477 IC50 = 2.2 nM T52450 CY0S2M 15851478 IC50 = 2.8 nM T52450 C2WHJ4 15859211 IC50 = 639 nM T52450 C5FA3L 15871222 IC50 = 104 nM T52450 CB3A4Z 15941413 Ki = 205000 nM T52450 CA40FE 15941550 Ki = 128000 nM T52450 CM3D1L 15941553 Ki = 5400 nM T52450 CQ0ZL7 15941677 Ki = 140000 nM T52450 C6R1LD 15985818 IC50 = 2471 nM T52450 CV67UL 15986261 IC50 = 557000 nM T52450 C4VW5F 16058482 IC50 = 35 nM T52450 C4WX2I 16108938 IC50 > 5000 nM T52450 CD51GI 16108939 IC50 = 3878 nM T52450 C5YVB0 16108940 IC50 > 5000 nM T52450 CB4DU9 16108941 IC50 > 5000 nM T52450 CBW71J 16108942 IC50 > 5000 nM T52450 CG6R9L 16108943 IC50 > 5000 nM T52450 CN62KM 16108944 IC50 > 5000 nM T52450 C7YS5Q 16108947 IC50 > 5000 nM T52450 CLD2Y4 16108948 IC50 > 5000 nM T52450 CJR95O 16108949 IC50 > 5000 nM T52450 CRQ26L 16108950 IC50 > 5000 nM T52450 CH80AG 16108951 IC50 = 2500 nM T52450 CWB0G9 16108952 IC50 > 5000 nM T52450 CS46XU 16126723 IC50 = 1530 nM T52450 C91EXN 16655061 IC50 = 2680 nM T52450 CQS0F5 16719301 IC50 > 10000 nM T52450 C75XDI 16730519 IC50 > 5000 nM T52450 C6F9LM 16748789 IC50 > 100000 nM T52450 C3S2TQ 17754305 IC50 = 5200 nM T52450 C6O3KA 17781194 IC50 = 280 nM T52450 CIR7S8 17866387 IC50 = 35 nM T52450 CL1H9W 17866459 IC50 = 142 nM T52450 C9RNH3 17866675 IC50 = 306 nM T52450 CCGR13 17897285 IC50 = 156 nM T52450 C2ZAX1 18002715 Ki > 4900 nM T52450 C12UGK 18002722 Ki > 4900 nM T52450 C0IYW8 18002726 Ki > 4900 nM T52450 C8N1DM 18002729 Ki > 4900 nM T52450 CCG96A 18002736 Ki > 4900 nM T52450 C5MLG1 18002745 Ki > 4900 nM T52450 CXT4H2 18002752 Ki > 4900 nM T52450 C26WHK 18002758 Ki > 4900 nM T52450 CV90XS 18002764 Ki > 4900 nM T52450 C8KPM7 18002765 Ki > 4900 nM T52450 CMJ0K3 18002771 Ki > 4900 nM T52450 C2CO9Z 18002775 Ki > 4900 nM T52450 CK8FS7 18173159 IC50 > 10000 nM T52450 CX10BM 18173179 IC50 = 2850 nM T52450 CQO70Y 18173222 IC50 > 1000 nM T52450 C6F8WH 18319167 IC50 = 8600 nM T52450 CXG1K2 18363133 IC50 > 10000 nM T52450 C37BNA 18363136 IC50 > 10000 nM T52450 C0KOW7 18363142 IC50 > 10000 nM T52450 CP04KS 18363146 IC50 > 10000 nM T52450 CLZD96 18363152 IC50 > 10000 nM T52450 CW3KB9 18363153 IC50 > 10000 nM T52450 CK30ZO 18363159 IC50 > 10000 nM T52450 CZU27R 18363164 IC50 > 10000 nM T52450 CC0UV8 18363169 IC50 > 10000 nM T52450 CR3CQ4 18363187 IC50 > 10000 nM T52450 CH5IU9 18363209 IC50 > 10000 nM T52450 CJGZ27 18363210 IC50 > 10000 nM T52450 CWI2A9 18363212 IC50 > 10000 nM T52450 C31LQZ 18363213 IC50 > 10000 nM T52450 CE60WD 18363216 IC50 > 10000 nM T52450 C3L6DU 18363223 IC50 > 10000 nM T52450 C6AW0H 18365436 IC50 = 100 nM T52450 C1QIU4 18368941 IC50 = 250000 nM T52450 C0VJG4 18368975 IC50 = 1500000 nM T52450 CI53DY 18379040 Ki > 4949 nM T52450 CB1U5T 18379077 Ki > 4949 nM T52450 CSX97G 18379115 Ki > 4949 nM T52450 CJHL25 18379123 Ki > 4949 nM T52450 CR0B8G 18379149 Ki > 4949 nM T52450 CS4V5K 18379187 Ki > 4949 nM T52450 CCTY94 18379210 Ki > 4949 nM T52450 CA6K5S 18379235 Ki > 4949 nM T52450 CCSK49 18379254 Ki > 4949 nM T52450 CP4T7S 18379435 Ki > 4949 nM T52450 C9Y5GX 18379443 Ki > 4949 nM T52450 CS2H6J 18396836 IC50 = 5000 nM T52450 C1WUJ0 18512732 IC50 = 40000 nM T52450 CA0JF9 18512733 IC50 = 300000 nM T52450 C8EIC6 18512737 IC50 > 10000000 nM T52450 C5B9WG 18533077 IC50 = 20000 nM T52450 CYA3H7 18790040 IC50 > 10000 nM T52450 CBN28Y 18790155 Ki > 10000 nM T52450 CRI35F 19366819 IC50 > 10000 nM T52450 CC4KN8 19366830 IC50 = 60 nM T52450 CS70KY 19366867 IC50 > 10000 nM T52450 CE73XW 19366873 IC50 > 10000 nM T52450 C60WKH 20196702 IC50 = 5616.56 nM T52450 CK8MP3 20620240 Ki > 10000 nM T52450 CPC4G6 20620273 Ki > 10000 nM T52450 C2E3CY 20620614 Ki = 5600 nM T52450 CPK09X 20651316 IC50 = 0.4 nM T52450 C30EAU 20651317 IC50 = 2117 nM T52450 CG1BD4 20689551 IC50 > 10000 nM T52450 C48TWB 20728102 IC50 > 5000 nM T52450 C18RXS 20735191 IC50 = 5900 nM T52450 C4I1OM 20735209 IC50 = 10000 nM T52450 CF1CK9 20735364 IC50 = 5000 nM T52450 CW3D7O 20760308 Ki > 4949 nM T52450 C09JTR 21130554 IC50 = 130 nM T52450 CW1JS2 21130555 IC50 > 10000000 nM T52450 C6VP1T 21130556 IC50 = 1200 nM T52450 C15UGO 21130558 IC50 > 10000 nM T52450 C9H3IG 21130559 IC50 = 1600 nM T52450 C8Q2OD 21130561 IC50 = 2400 nM T52450 C25FAD 21130562 IC50 = 700 nM T52450 C3FAU5 21130572 IC50 = 400000 nM T52450 C19AEV 21130574 IC50 = 600000 nM T52450 CW2Q5A 21130590 IC50 > 10000 nM T52450 C9HMC0 21130591 IC50 > 10000 nM T52450 CM92DX 21304705 IC50 = 226 nM T52450 CJ0Y9V 21304706 IC50 = 92 nM T52450 C5X1YM 21304708 IC50 = 6 nM T52450 C0Z3LD 21304710 IC50 = 1 nM T52450 CG18HB 21310751 IC50 = 470 nM T52450 CEW0M3 21310753 IC50 = 213 nM T52450 C0T2QX 21310757 IC50 = 291 nM T52450 CWM7F2 21310775 IC50 = 520 nM T52450 CNEW70 21310777 IC50 = 115 nM T52450 CY12PI 21310778 IC50 = 202 nM T52450 CPT4E5 21310780 IC50 = 884 nM T52450 CJ2U7K 21310781 IC50 = 553 nM T52450 C5SG2L 21310789 IC50 = 744 nM T52450 C3TI6Y 21310790 IC50 = 18 nM T52450 C87BMF 21310824 IC50 = 608 nM T52450 C26IPQ 21310829 IC50 = 132 nM T52450 CIB1X5 21310851 IC50 = 781 nM T52450 C6OZL3 21310926 IC50 = 1050 nM T52450 C72BVA 21310934 IC50 = 1573 nM T52450 C96REO 21584504 IC50 = 82 nM T52450 CT87YK 21699971 IC50 > 10000000 nM T52450 CH4G5T 21699977 IC50 > 50000 nM T52450 CQ1GI3 21699983 IC50 = 14000000 nM T52450 CJZ58F 21699985 IC50 > 10000000 nM T52450 CA3WG1 21699989 IC50 > 10000 nM T52450 CE72FU 21700004 IC50 > 10000000 nM T52450 CRG8J9 21700008 IC50 = 840 nM T52450 C5JC6W 21700038 IC50 = 4100000 nM T52450 CY18IE 21700054 IC50 = 1100 nM T52450 CW1YS9 21700072 IC50 = 1600 nM T52450 C3QAP8 21700080 IC50 > 10000000 nM T52450 CR81NU 21700137 IC50 > 10000 nM T52450 CJ4C3K 21700144 IC50 = 1600 nM T52450 C94FZS 21700146 IC50 > 10000 nM T52450 CXME27 21700151 IC50 = 4200000 nM T52450 CFK4Y7 21700160 IC50 = 14000000 nM T52450 CIJ93L 21700163 IC50 = 360000 nM T52450 CN80JR 21700178 IC50 = 440 nM T52450 CB1QH3 21700191 IC50 > 10000000 nM T52450 CUVE24 21700204 IC50 > 10000000 nM T52450 CM42ZR 21700258 IC50 > 10000 nM T52450 CMW12T 21700264 IC50 = 1000 nM T52450 C45UGA 21996090 IC50 > 10000 nM T52450 CIC4S9 22004232 IC50 = 920 nM T52450 C36WFA 22096205 IC50 > 100000 nM T52450 CH6U1G 22338710 IC50 = 747 nM T52450 CO91AD 22341241 Ki > 4949 nM T52450 CN04BS 22463223 Ki = 33 nM T52450 CZT05X 22484417 Ki > 10000 nM T52450 CZT64B 22484431 Ki > 10000 nM T52450 C1O7RC 22485248 IC50 > 10000 nM T52450 CAM10T 22485252 IC50 > 10000 nM T52450 CBJS34 22485260 IC50 = 2500 nM T52450 CEGJ03 22485276 IC50 > 10000 nM T52450 C7VB8G 22485289 IC50 = 1000 nM T52450 CNB02I 22485291 IC50 = 300 nM T52450 CAY3N6 22485292 IC50 > 10000 nM T52450 C94OCJ 22485302 IC50 = 1000 nM T52450 C3YL5X 22485311 IC50 > 10000 nM T52450 C80RSQ 22485314 IC50 = 10000 nM T52450 CWA03L 22485327 IC50 = 4500 nM T52450 C6JRW5 22485340 IC50 = 770 nM T52450 C5JZF1 22485344 IC50 = 3600 nM T52450 CI7MY5 22485346 IC50 = 1400 nM T52450 CI1YL7 22485347 IC50 = 2400 nM T52450 C25OBD 22485356 IC50 = 1800 nM T52450 C7I0EW 22485367 IC50 = 400 nM T52450 CL64TJ 22485368 IC50 > 10000 nM T52450 CT4GF9 22485381 IC50 > 10000 nM T52450 C27NDB 22485386 IC50 > 10000 nM T52450 CTJ9I3 22485392 IC50 = 2000 nM T52450 C3MG9P 22485396 IC50 = 4400 nM T52450 CZY10U 22485408 IC50 > 10000 nM T52450 C89AGT 22485413 IC50 = 2000 nM T52450 C03NLM 22485417 IC50 = 268 nM T52450 C8GHU9 22485432 IC50 = 6000 nM T52450 C5TB0U 22615571 IC50 = 360 nM T52450 CP2J9V 22615653 Ki = 423 nM T52450 C9BT5F 22626996 IC50 = 7250 nM T52450 C7ITG0 22644780 IC50 = 238 nM T52450 CIQ76F 22644837 IC50 = 92 nM T52450 CYJ48I 22644895 IC50 = 408 nM T52450 CQB36V 22644965 IC50 = 113 nM T52450 CVM1O6 22644970 IC50 = 287 nM T52450 C0K1GE 22645081 IC50 = 1156 nM T52450 C2Q4XK 22707806 IC50 = 3600 nM T52450 CMYK90 22707860 IC50 = 4500 nM T52450 CVF9M4 22922043 IC50 = 10560 nM T52450 COCN69 22956916 Ki > 4949 nM T52450 C85PXN 22956934 Ki > 4949 nM T52450 CIYA45 22985930 IC50 = 10000 nM T52450 CM5H2P 23061661 IC50 > 10000 nM T52450 C97LAR 23061665 IC50 > 10000 nM T52450 C9IW3E 23433373 IC50 > 10000 nM T52450 C4VG8C 23506747 IC50 = 1534 nM T52450 CK97AT 23506779 IC50 = 2488 nM T52450 CP94QR 23506783 IC50 = 114 nM T52450 CX32YK 23513795 IC50 = 2700 nM T52450 C6IZ1S 23513821 IC50 = 6270 nM T52450 CPNM93 23513825 IC50 = 3040 nM T52450 CML90Q 23513831 IC50 = 3320 nM T52450 C8UIC6 23644662 Ki > 100000 nM T52450 CCLA40 23644663 Ki > 100000 nM T52450 CSZ6J4 23645528 IC50 = 25.7 nM T52450 C6UH9Q 23645529 Ki = 7 nM T52450 CD0JP3 23645530 Ki = 7 nM T52450 CM37EC 23645531 IC50 = 20.89 nM T52450 C9PD5F 23645532 IC50 = 23.99 nM T52450 C1OE7R 23645533 IC50 = 6.918 nM T52450 CCSN04 23645534 Ki = 60 nM T52450 CU08WI 23645535 IC50 = 3.981 nM T52450 CY41UC 23645536 Ki = 25 nM T52450 CX15EH 23645537 Ki = 37 nM T52450 CD3Q6G 23645538 IC50 = 52.48 nM T52450 CE6NQ2 23645539 Ki = 74000 nM T52450 C4VK3U 23645540 Ki = 70000 nM T52450 C8VM1C 23645541 Ki = 95000 nM T52450 C0MUT6 23645542 Ki = 42000 nM T52450 CNI07H 23645543 Ki = 37000 nM T52450 CHK2X1 23645544 Ki = 59000 nM T52450 CW1V2Z 23645545 Ki = 30000 nM T52450 C6SP7T 23645546 Ki = 30000 nM T52450 CD9QO2 23645547 Ki = 400 nM T52450 C25YLZ 23645548 Ki = 80 nM T52450 C4R2DA 23645953 Ki > 300000 nM T52450 CWN3I4 23645959 Ki > 300000 nM T52450 CL1KC0 23652834 IC50 = 3219.85 nM T52450 C6AW7U 23692637 IC50 = 25000 nM T52450 C7KF1N 23729138 IC50 = 250000 nM T52450 C3TWS6 24178109 Ki = 67 nM T52450 CY6KA0 24755074 IC50 = 25000 nM T52450 CQCJ17 24768595 IC50 > 1000 nM T52450 C5M3YW 24799779 Ki > 10000000 nM T52450 CWLT01 24806172 IC50 > 10000 nM T52450 CN59KZ 24806173 IC50 > 10000 nM T52450 CH4X8K 24806175 IC50 > 10000 nM T52450 C18FRG 24807817 IC50 = 90000 nM T52450 CW3X0F 24852010 IC50 > 1000 nM T52450 C6YPS8 24852048 IC50 > 1000 nM T52450 C4UEM5 24871537 Ki > 50000 nM T52450 CP2L5B 24871655 Ki > 50000 nM T52450 CFL04M 24881245 IC50 > 300000 nM T52450 CLIC14 24881246 IC50 = 270000 nM T52450 C02WIB 24882535 IC50 > 10000 nM T52450 C4FI5C 24901479 IC50 = 5400 nM T52450 C4SP3O 24936157 IC50 = 170 nM T52450 CBUA83 24936183 IC50 > 1000 nM T52450 CQ2K9H 24936215 IC50 > 5000 nM T52450 CH3O0V 24951588 IC50 > 10000 nM T52450 C8I4PT 24951589 IC50 > 10000 nM T52450 C2Q1BK 24951590 IC50 > 10000 nM T52450 COMJ45 24951950 IC50 > 10000 nM T52450 C3JGU2 24951952 IC50 > 10000 nM T52450 CC7U2T 24951953 IC50 > 10000 nM T52450 CV86KA 24952316 IC50 > 10000 nM T52450 CYKM71 24952674 IC50 > 10000 nM T52450 C7MC8J 24952678 IC50 > 10000 nM T52450 C5BG6I 24955154 IC50 > 10000 nM T52450 CCE45B 24955155 IC50 > 10000 nM T52450 CH53AG 24955156 IC50 > 10000 nM T52450 CZC1P7 24955511 IC50 > 10000 nM T52450 CXO9Y4 24955857 IC50 > 10000 nM T52450 C4LJ8N 24955859 IC50 > 10000 nM T52450 CX4MY3 24955861 IC50 > 10000 nM T52450 CR29SO 24956227 IC50 > 10000 nM T52450 CSM26P 24956228 IC50 > 10000 nM T52450 C13JHO 24956229 IC50 > 10000 nM T52450 C01QMC 24956580 IC50 > 10000 nM T52450 C8M5PJ 24956581 IC50 > 10000 nM T52450 CC90AR 24956582 IC50 > 10000 nM T52450 CQH6I4 24956585 IC50 > 10000 nM T52450 CHJ50Q 24956943 IC50 > 10000 nM T52450 CN2AS5 24956945 IC50 > 10000 nM T52450 C2HN8M 24956948 IC50 > 10000 nM T52450 CNCA57 25004194 Ki > 5000 nM T52450 CAQ9Z1 25022681 Ki > 4946 nM T52450 CA86UE 25049752 Ki = 143 nM T52450 C82NLV 25049754 Ki = 151 nM T52450 C6QFV4 25049756 Ki = 3400 nM T52450 CVR52U 25066764 IC50 > 6 nM T52450 CD2KA4 25102047 IC50 = 780 nM T52450 CRW96X 25102048 IC50 = 320 nM T52450 CQ3O9P 25102050 IC50 = 280 nM T52450 CSHA26 25102051 IC50 = 1300 nM T52450 C7ADO2 25102197 IC50 = 1400 nM T52450 CA5DJ4 25138228 Ki > 10000000 nM T52450 C1TNQ3 25141117 IC50 = 30 nM T52450 CR35QP 25144971 IC50 > 10000 nM T52450 C0Y5BC 25145683 IC50 > 2500 nM T52450 CB7V8Y 25147773 IC50 = 7.8 nM T52450 C3KF1V 25178145 IC50 = 143 nM T52450 CG5Y2R 25178357 IC50 = 236 nM T52450 C4PZY6 25180866 IC50 = 235 nM T52450 CEP9Q2 25180867 IC50 = 59 nM T52450 C7U1YC 25181080 IC50 = 532 nM T52450 C85HLG 25181081 IC50 = 542 nM T52450 CHR2P1 25183768 Ki > 25000 nM T52450 CZ8CR1 25190501 Ki > 4948 nM T52450 CO8CD1 25190502 Ki > 4948 nM T52450 C9GCO4 28602444 IC50 > 150000 nM T52450 C0H3RD 42627769 IC50 > 50000 nM T52450 CPO1Z3 44123600 IC50 = 4540 nM T52450 C9LF6X 44143582 IC50 = 3350 nM T52450 CIH43B 44143583 IC50 > 10000 nM T52450 CRO9K7 44143584 IC50 > 10000 nM T52450 CNT3R8 44143585 IC50 = 3600 nM T52450 C9TXG7 44143586 IC50 > 10000 nM T52450 CYW27E 44143587 IC50 > 10000 nM T52450 C7XOT1 44143588 IC50 > 10000 nM T52450 CQ2RN8 44143589 IC50 > 10000 nM T52450 CF40SE 44143590 IC50 > 10000 nM T52450 CE7X2W 44143600 IC50 > 10000 nM T52450 CYJ0Z4 44143601 IC50 = 3230 nM T52450 CP1UO5 44143602 IC50 = 680 nM T52450 CP8L7N 44143603 IC50 = 950 nM T52450 CRL6C0 44143605 IC50 > 10000 nM T52450 C09OTR 44143606 IC50 > 10000 nM T52450 CTM85Q 44143607 IC50 > 10000 nM T52450 CV8BO6 44143608 IC50 = 2020 nM T52450 C8HR2I 44143609 IC50 = 6370 nM T52450 C90ISP 44143610 IC50 > 10000 nM T52450 C2J5IT 44143611 IC50 > 10000 nM T52450 CO9N4R 44143612 IC50 = 9330 nM T52450 C85DBI 44143613 IC50 > 10000 nM T52450 CQZ2W1 44143614 IC50 > 10000 nM T52450 CAP7M2 44143615 IC50 > 10000 nM T52450 C3DX9H 44143616 IC50 > 10000 nM T52450 CIY4K3 44143617 IC50 > 10000 nM T52450 CRQ0T5 44143618 IC50 = 7050 nM T52450 COP5G1 44143619 IC50 = 1740 nM T52450 CM45NB 44143620 IC50 = 1290 nM T52450 C20COZ 44143621 IC50 = 770 nM T52450 CZC0U7 44143622 IC50 = 6560 nM T52450 CR4ZF1 44143623 IC50 = 2300 nM T52450 CZU83Q 44143624 IC50 = 4180 nM T52450 CS26DC 44143625 IC50 > 10000 nM T52450 C8B3VE 44143626 IC50 > 10000 nM T52450 CG78RF 44143627 IC50 > 10000 nM T52450 C8VQS4 44143628 IC50 > 10000 nM T52450 CKV3C6 44143629 IC50 = 4300 nM T52450 CK21NW 44143630 IC50 = 650 nM T52450 C4ELQ8 44143631 IC50 = 12900 nM T52450 C9S8YH 44143632 IC50 > 10000 nM T52450 CCZP24 44143633 IC50 > 10000 nM T52450 C3VBX4 44143634 IC50 > 10000 nM T52450 CU02HY 44143635 IC50 > 10000 nM T52450 C16VZT 44143636 IC50 > 10000 nM T52450 CSQ0V9 44143637 IC50 > 10000 nM T52450 C27UYE 44143638 IC50 > 10000 nM T52450 C5K2OM 44143639 IC50 > 10000 nM T52450 CI7H6E 44143640 IC50 > 10000 nM T52450 CT80ED 44219901 IC50 = 13000 nM T52450 C94JVY 44219902 IC50 = 5600 nM T52450 C7J6GH 44219903 IC50 = 59000 nM T52450 C9J7WL 44219904 IC50 = 13000 nM T52450 CRQ71E 44219905 IC50 = 20000 nM T52450 C4Z0ID 44219906 IC50 > 10000 nM T52450 CRNA25 44220092 IC50 > 10000 nM T52450 C9T5ZF 44220093 IC50 = 48000 nM T52450 CV38TE 44222825 IC50 = 11000 nM T52450 CJI73R 44222826 IC50 = 3300 nM T52450 CGQ30N 44222827 IC50 = 13000 nM T52450 CCI64J 44224245 IC50 = 5460 nM T52450 CLRT69 44247751 IC50 = 3500 nM T52450 CAR34Y 44263877 IC50 = 2200 nM T52450 CEV08N 44263913 IC50 = 97 nM T52450 C5ZI0X 44263926 IC50 = 13.6 nM T52450 CO3C1E 44263994 IC50 = 346 nM T52450 C9XJ7U 44264020 IC50 = 696 nM T52450 C6L0MJ 44264021 IC50 = 22 nM T52450 CJ1WE7 44264036 IC50 = 465 nM T52450 C50QFR 44264375 IC50 = 643 nM T52450 CDL25C 44265349 Ki > 5000 nM T52450 C3W4QO 44265401 Ki > 5000 nM T52450 C2Q3JV 44265407 Ki = 4868 nM T52450 CN59QT 44265437 Ki > 5000 nM T52450 CZA61K 44265475 Ki > 5000 nM T52450 CD4A7F 44265476 Ki > 5000 nM T52450 CT6FK0 44265480 Ki = 4107 nM T52450 C67HUL 44265485 Ki > 5000 nM T52450 CH0O3I 44265492 Ki > 5000 nM T52450 C0DFG7 44265501 Ki > 5000 nM T52450 CXSD62 44265506 Ki > 10000 nM T52450 CCM8K0 44265512 Ki = 1931 nM T52450 CB3E6O 44265527 Ki = 1820 nM T52450 COU3Y8 44266817 IC50 = 4200 nM T52450 CUA5E0 44266818 IC50 = 3400 nM T52450 CG23BI 44266830 IC50 > 10000 nM T52450 C3HP1F 44270658 IC50 > 20 nM T52450 C8S2FJ 44270678 IC50 = 1300 nM T52450 C2BUH0 44270679 IC50 > 20 nM T52450 C4C3RN 44270683 IC50 = 1700 nM T52450 C4OJK9 44270703 IC50 = 430 nM T52450 C8MUJ3 44270704 IC50 > 10 nM T52450 C7CVT3 44270713 IC50 = 200 nM T52450 C0K3RP 44270736 IC50 = 1500 nM T52450 CLMO84 44270737 IC50 = 69 nM T52450 CKL2C3 44270739 IC50 > 10 nM T52450 C4B0LP 44270775 IC50 > 10 nM T52450 CYZX59 44270776 IC50 > 20 nM T52450 C1WTN7 44270802 IC50 = 1500 nM T52450 C6UQ8N 44270804 IC50 = 380 nM T52450 CVG61X 44270805 IC50 = 890 nM T52450 CNU41R 44270901 IC50 > 10000 nM T52450 CDX36Y 44270985 IC50 > 4000 nM T52450 CFR81A 44271005 IC50 = 140 nM T52450 CRF2Z5 44271421 IC50 = 3235.42 nM T52450 CG92WS 44272353 IC50 = 1658 nM T52450 CO2Z6K 44272475 IC50 = 194 nM T52450 C63KSL 44272540 IC50 = 1923 nM T52450 CG7X5F 44272675 IC50 = 15 nM T52450 C20JLP 44272837 IC50 > 30000 nM T52450 CEHR24 44272853 IC50 = 3.5 nM T52450 C4YM6S 44272911 IC50 > 30000 nM T52450 C6ON3U 44273235 IC50 > 30000 nM T52450 CV6T9M 44273670 Ki = 15900 nM T52450 C2RA8T 44273710 Ki = 5100 nM T52450 C4SHN1 44273711 Ki = 2900 nM T52450 CO79TR 44273726 Ki = 7500 nM T52450 CGS86N 44275415 IC50 = 270 nM T52450 C02CJL 44275451 IC50 = 7400 nM T52450 CLV8N9 44275503 IC50 = 15000 nM T52450 CRD42Q 44275504 IC50 = 1900 nM T52450 CU95DJ 44275512 IC50 = 4500 nM T52450 C36TMQ 44275540 IC50 = 2200 nM T52450 CE3FT4 44275593 IC50 = 11000 nM T52450 CSJ50I 44275605 IC50 = 45 nM T52450 CQL60W 44275699 IC50 = 750 nM T52450 C5IMT1 44275731 IC50 = 20000 nM T52450 CKG24Z 44275742 IC50 = 18000 nM T52450 C8CB4A 44275752 IC50 = 690 nM T52450 CW3TX0 44275753 IC50 = 2300 nM T52450 CVI56W 44275768 IC50 = 22000 nM T52450 CV3IQ8 44275769 IC50 = 60 nM T52450 C1O4TU 44275790 IC50 = 19000 nM T52450 CV2WC5 44275791 IC50 = 1800 nM T52450 CUD36E 44275806 IC50 = 180 nM T52450 CPXV83 44275825 IC50 = 200 nM T52450 CZJ0U5 44275897 IC50 = 2800 nM T52450 CG0H1Q 44275898 IC50 = 1700 nM T52450 CMU92H 44275912 IC50 = 2100 nM T52450 CB6SM0 44275938 IC50 = 5100 nM T52450 CZK8S5 44275954 IC50 > 30000 nM T52450 CIK26Z 44276134 IC50 = 3500 nM T52450 CTO6V2 44278377 IC50 = 1600 nM T52450 C2Z6MF 44278411 IC50 = 12000 nM T52450 C9X8DM 44278412 IC50 = 6500 nM T52450 CJ8ON1 44278424 IC50 = 16000 nM T52450 CEA0H3 44278449 IC50 = 3000 nM T52450 CC4V8G 44278484 IC50 = 30000 nM T52450 CJ78PR 44278512 IC50 = 23000 nM T52450 C1GLP0 44278522 IC50 = 5800 nM T52450 CAB1C5 44278523 IC50 = 3700 nM T52450 C04WHR 44278532 IC50 = 30000 nM T52450 CK16OS 44278550 IC50 = 24000 nM T52450 CJ94UF 44278576 IC50 = 8.5 nM T52450 CQDI85 44278667 IC50 = 19 nM T52450 C6YT3K 44280285 Ki = 432 nM T52450 C8XUJ3 44280321 Ki = 20 nM T52450 CC2O3U 44280323 Ki = 5 nM T52450 CM2TZ4 44280335 Ki = 2.3 nM T52450 CIE09F 44280336 Ki = 3 nM T52450 CA1V6Y 44280345 Ki = 1 nM T52450 CI9L2E 44280411 Ki = 171 nM T52450 C87WBN 44280461 Ki = 1500 nM T52450 C8KZ2F 44281541 IC50 = 37 nM T52450 CRK8H6 44281557 IC50 = 52 nM T52450 CTJ7Q2 44281563 IC50 = 2.7 nM T52450 COU71D 44281564 IC50 = 110 nM T52450 CJ2PG9 44281705 IC50 = 6.9 nM T52450 CC2QR7 44281720 Ki = 440 nM T52450 C1M3JR 44281777 IC50 = 50 nM T52450 CL18QW 44281786 IC50 = 120 nM T52450 C3ES4Z 44281796 IC50 = 1.3 nM T52450 C60HIN 44281797 IC50 = 9.4 nM T52450 C8U5GR 44281941 IC50 = 550 nM T52450 CN23FC 44282968 IC50 = 25000 nM T52450 C2TV5I 44282969 IC50 = 20000 nM T52450 CG3LF0 44282970 IC50 > 30000 nM T52450 C6S3GN 44283598 IC50 = 200 nM T52450 CXE73H 44283613 IC50 = 1922 nM T52450 CP3L2U 44283938 IC50 = 177 nM T52450 C6JLI2 44285620 Ki = 16000 nM T52450 CC5XL3 44286083 IC50 = 4900 nM T52450 CXT37W 44286406 IC50 > 50000 nM T52450 CB1R9G 44286414 IC50 > 10000 nM T52450 C7CU3J 44286466 IC50 = 2500000 nM T52450 CZ2AL1 44286483 IC50 > 50000 nM T52450 C8I2EF 44286485 IC50 > 10000 nM T52450 C48FEB 44286518 IC50 = 3600 nM T52450 CKM8V6 44286563 IC50 > 10000 nM T52450 C3UB9V 44286654 Ki > 850 nM T52450 CB07MX 44286663 Ki = 552.4 nM T52450 C3KXY9 44286674 Ki = 90 nM T52450 C96NMF 44287796 IC50 = 3500 nM T52450 CQ5IG7 44287805 IC50 = 40 nM T52450 CHOV34 44287806 IC50 = 9 nM T52450 CYAG29 44287899 IC50 = 29 nM T52450 CX5QB3 44287917 IC50 = 7 nM T52450 CCM31I 44288043 IC50 = 6 nM T52450 C1YT7H 44288071 IC50 = 22 nM T52450 CF2DZ9 44288091 IC50 = 480 nM T52450 CMY2N4 44288092 IC50 = 170 nM T52450 CCS20R 44288093 IC50 = 3 nM T52450 CJ1HT6 44288855 IC50 > 10000 nM T52450 CT38HI 44289140 IC50 > 10000 nM T52450 CAH30U 44289181 IC50 > 10000 nM T52450 CH1TS5 44289182 IC50 > 10000 nM T52450 CMZ2O6 44289200 IC50 > 10000 nM T52450 CBLC60 44289352 Ki = 9590 nM T52450 CZO75J 44289369 Ki = 1010 nM T52450 CRT7O2 44289382 Ki = 1710 nM T52450 C7WUJ2 44289459 IC50 > 10000 nM T52450 CJ73FW 44289479 IC50 > 10000 nM T52450 CWMI67 44289482 IC50 > 10000 nM T52450 C1L4ZU 44289489 IC50 > 10000 nM T52450 C19EJM 44289515 IC50 > 10000 nM T52450 C6TI3X 44289520 Ki > 10000 nM T52450 CA52ED 44289521 Ki > 10000 nM T52450 C30KSP 44289579 Ki > 10000 nM T52450 CHC08W 44289601 Ki = 400 nM T52450 CZ4EI7 44289602 Ki = 1710 nM T52450 CEML82 44289603 Ki = 1900 nM T52450 CM26JT 44289604 Ki = 1720 nM T52450 CLY4K5 44289640 Ki = 357 nM T52450 C7GY8M 44289643 Ki > 10000 nM T52450 CV9B2F 44289867 Ki > 10000 nM T52450 CO9V6X 44291148 IC50 = 41200 nM T52450 CJ7VW3 44291166 IC50 = 104 nM T52450 C30EAH 44291219 IC50 = 37000 nM T52450 C2SNP3 44291220 IC50 = 3460 nM T52450 CT83ZH 44291511 IC50 > 10000 nM T52450 CYS89X 44291521 IC50 = 2900 nM T52450 CF21CS 44291532 IC50 = 156 nM T52450 CB02YN 44291538 IC50 = 15700 nM T52450 CU75TB 44291559 IC50 = 384 nM T52450 C8CV6U 44291796 IC50 = 350 nM T52450 CCDP84 44292860 IC50 = 460 nM T52450 CG39PV 44292881 IC50 = 3800 nM T52450 CAT41C 44292981 IC50 = 800 nM T52450 CQ2E1B 44292992 IC50 = 770 nM T52450 CV5ID4 44293016 IC50 = 17500 nM T52450 C0B9AI 44293038 IC50 = 40 nM T52450 CRAK57 44293116 IC50 = 570 nM T52450 C9NOK3 44293155 IC50 = 90 nM T52450 CPRT90 44293156 IC50 = 23 nM T52450 C3IGW2 44293230 IC50 = 140 nM T52450 CJ47YX 44293231 IC50 = 260 nM T52450 C9HX1S 44293286 IC50 = 2800 nM T52450 CV0Y8U 44293304 IC50 = 3200 nM T52450 C3UKB6 44293306 IC50 > 30000 nM T52450 CL4F5R 44293307 IC50 = 570 nM T52450 C4LI6F 44293416 Ki = 0.87 nM T52450 CVA3H0 44293739 IC50 = 140 nM T52450 CZ1L4M 44293821 IC50 = 12000 nM T52450 CWD36G 44293839 IC50 = 3000 nM T52450 CW7Z5H 44293865 IC50 > 30000 nM T52450 C5XS0I 44294322 Ki = 2860 nM T52450 CC4V8S 44295180 IC50 = 60 nM T52450 CRW07Z 44295181 IC50 = 6 nM T52450 CL5QG6 44295202 IC50 = 860 nM T52450 CF0T8W 44295423 IC50 = 730 nM T52450 CVS7I1 44295425 IC50 = 50 nM T52450 CAFB18 44296974 Ki > 4949 nM T52450 C8NTY1 44299442 IC50 = 147 nM T52450 CE34KO 44299443 IC50 = 171 nM T52450 C7Z0IF 44299460 IC50 = 130 nM T52450 C06NTZ 44299503 IC50 = 105 nM T52450 C8E0UV 44299522 IC50 = 5000 nM T52450 CQSA71 44299538 IC50 = 93 nM T52450 C69TNW 44299709 IC50 > 100000 nM T52450 C2LXS8 44299719 IC50 = 26 nM T52450 C3ASF8 44299722 IC50 = 7000 nM T52450 CNHR69 44299733 IC50 = 4000 nM T52450 C03HUT 44299735 IC50 = 8 nM T52450 CI9GR7 44299736 IC50 = 4000 nM T52450 C6HY7N 44299870 IC50 = 83 nM T52450 COV3W7 44299871 IC50 = 3498 nM T52450 C9R2FL 44299872 IC50 = 598 nM T52450 CTGR41 44299873 IC50 = 425 nM T52450 C8K6VC 44299880 IC50 = 215 nM T52450 C2WZ7S 44299893 IC50 = 250 nM T52450 CG3EJ5 44299894 IC50 = 40 nM T52450 CD5Y6C 44299895 IC50 = 63 nM T52450 CA5EN9 44299909 IC50 = 453 nM T52450 CRDX61 44299910 IC50 = 26 nM T52450 C79UQM 44299911 IC50 = 12 nM T52450 C6PDF1 44299928 IC50 = 34 nM T52450 C5RSX9 44300181 IC50 = 58000 nM T52450 CKN3P7 44302022 IC50 = 5000 nM T52450 C2Y0PK 44302023 IC50 = 4130 nM T52450 C5S3UO 44302024 IC50 = 4730 nM T52450 C8ERW6 44302042 IC50 = 5960 nM T52450 C6JXH0 44302043 IC50 = 7943.28 nM T52450 CWB83G 44302076 IC50 = 4110 nM T52450 CY1J9U 44302096 IC50 = 4183 nM T52450 CW94ZQ 44302164 IC50 = 8950 nM T52450 C2FSR6 44302165 IC50 = 375 nM T52450 CQ54PZ 44302166 IC50 = 300 nM T52450 C9U3XT 44302167 IC50 = 5000 nM T52450 C5X1WY 44302183 IC50 = 6728 nM T52450 CQS19O 44302187 IC50 = 20000 nM T52450 C7G3BN 44302200 IC50 = 4999 nM T52450 C70QWV 44302327 IC50 = 19952.62 nM T52450 CZP20C 44302339 IC50 = 9829 nM T52450 CO73BW 44302357 IC50 = 3780 nM T52450 CXUZ19 44302359 IC50 = 50000 nM T52450 C6YB0Q 44302364 IC50 = 7000 nM T52450 CCW65Y 44302378 IC50 = 20 nM T52450 CYG80V 44302385 IC50 = 1000 nM T52450 C7ZBR4 44302396 IC50 = 150 nM T52450 C8S5WT 44302397 IC50 = 400 nM T52450 CPC25G 44302409 IC50 = 5370 nM T52450 C4QL0I 44302411 IC50 = 500 nM T52450 C4NDA2 44302416 IC50 = 8270 nM T52450 C24ZWF 44302429 IC50 = 4660 nM T52450 C4I6WO 44302430 IC50 = 3000 nM T52450 CYL71W 44302432 IC50 = 3019.95 nM T52450 C5H6OV 44302627 IC50 = 4350 nM T52450 C6QR7C 44302634 IC50 = 7960 nM T52450 CG8KJ0 44302661 IC50 = 2190 nM T52450 CUZS20 44302663 IC50 = 7000 nM T52450 CX1M3Q 44302666 IC50 = 5350 nM T52450 C36CQP 44302952 IC50 = 7910 nM T52450 CPHG53 44302959 IC50 = 2153 nM T52450 CLMW26 44302960 IC50 = 1273 nM T52450 CRI6M5 44302961 IC50 = 1223 nM T52450 CLP1N4 44303118 IC50 = 6259 nM T52450 CYBZ65 44303119 IC50 = 1938 nM T52450 CP58IJ 44303125 IC50 = 5030 nM T52450 CK7EZ5 44303126 IC50 = 110 nM T52450 CG1XV5 44303128 IC50 = 6032 nM T52450 C7S6CJ 44303135 IC50 = 3271 nM T52450 C3AJ5R 44303143 IC50 = 823 nM T52450 CVA4U2 44303153 IC50 = 680 nM T52450 C6NK2T 44303154 IC50 = 2933 nM T52450 C9WMT6 44303156 IC50 = 669 nM T52450 CJ5H1N 44303159 IC50 = 1059 nM T52450 CJ9DX7 44303160 IC50 = 739 nM T52450 CJ17AT 44303161 IC50 = 135 nM T52450 CDM8U9 44303162 IC50 = 3473 nM T52450 CEG23F 44303163 IC50 = 953 nM T52450 CW7FB9 44303168 IC50 = 700 nM T52450 C39BFH 44303186 IC50 > 10000 nM T52450 C3GZX1 44303187 IC50 = 1330 nM T52450 CVY62P 44303199 IC50 = 5909 nM T52450 CP7TV3 44303235 IC50 = 561 nM T52450 CALD50 44304020 Ki > 5000 nM T52450 CTU4S6 44304048 Ki = 2238 nM T52450 C0IJ9D 44304112 Ki = 40.4 nM T52450 CSVK45 44304230 Ki > 5000 nM T52450 C7ME6Z 44305408 IC50 = 96 nM T52450 CD9W5Q 44305414 IC50 = 49 nM T52450 CY18UG 44305656 IC50 = 1890 nM T52450 C4QIF8 44305668 IC50 = 140 nM T52450 CA0GN1 44305669 IC50 = 117 nM T52450 CNF86G 44305670 IC50 = 57 nM T52450 CXF6Y3 44305706 IC50 = 3900 nM T52450 CCHK59 44305722 IC50 = 129 nM T52450 C6EZU9 44305732 IC50 = 225 nM T52450 C4ZI6D 44305743 IC50 = 51 nM T52450 CI82ZH 44305746 IC50 = 112 nM T52450 CLK31H 44305747 IC50 = 4360 nM T52450 COI82F 44305750 IC50 = 83 nM T52450 CLH14M 44305978 IC50 = 2.2 nM T52450 CZ49UN 44305988 IC50 = 2.1 nM T52450 C6I8JA 44306058 IC50 = 3 nM T52450 CB5EY3 44306200 IC50 = 6.6 nM T52450 C0YOH1 44306202 IC50 = 2.7 nM T52450 CMA39E 44306203 IC50 = 4.6 nM T52450 CL58OS 44306208 IC50 > 10000 nM T52450 CAY2S4 44306209 IC50 = 1400 nM T52450 C27NJX 44306277 IC50 = 210 nM T52450 C6O1AN 44306279 IC50 = 6.1 nM T52450 C5QUK2 44308295 Ki = 170 nM T52450 C2E4IT 44308297 Ki = 36 nM T52450 C0K4UQ 44308298 Ki = 41 nM T52450 CCRW50 44308304 Ki = 97 nM T52450 CZF5S2 44308327 Ki = 47 nM T52450 COE56H 44308377 Ki = 17 nM T52450 C7OT6S 44308488 Ki = 181 nM T52450 CI2Z0H 44308525 Ki = 16 nM T52450 CU0J5A 44308623 Ki = 55 nM T52450 CSEB94 44308624 Ki = 42 nM T52450 CST39W 44308640 Ki = 27 nM T52450 C5AM6P 44308844 IC50 = 5769.78 nM T52450 C4SJF3 44309329 IC50 = 745 nM T52450 C7ED1H 44309330 IC50 = 542 nM T52450 C1E3KF 44309437 IC50 = 195 nM T52450 C6N5SL 44309531 IC50 = 2268 nM T52450 CJ0L4P 44309550 IC50 = 1314 nM T52450 CKEU31 44309629 IC50 = 319 nM T52450 C6J3WN 44309662 IC50 = 103 nM T52450 CY96UH 44309686 IC50 = 376 nM T52450 CWNX29 44309720 IC50 = 2000 nM T52450 CMW0U4 44309879 IC50 = 74 nM T52450 CK6BT0 44309901 IC50 = 4640 nM T52450 C5I2AD 44310338 IC50 = 10000 nM T52450 C0B4HZ 44312333 IC50 = 38.9 nM T52450 CK9XB7 44314087 IC50 = 8300 nM T52450 C8MRB1 44314322 IC50 > 50000 nM T52450 CB6UL7 44314349 IC50 > 50000 nM T52450 C3R0DL 44314366 IC50 > 50000 nM T52450 C5ZTU6 44314442 Ki = 100000 nM T52450 C2JUX9 44314443 Ki = 41400 nM T52450 C92MGV 44314566 IC50 = 82 nM T52450 CLT6E0 44314618 IC50 = 4600 nM T52450 CC95EZ 44314744 Ki = 7.8 nM T52450 CY63DG 44314754 Ki = 302 nM T52450 C8ZD7F 44314755 Ki = 20892.96 nM T52450 COF0B1 44314762 Ki = 921 nM T52450 C59CBZ 44314763 Ki = 203 nM T52450 C9L1NY 44314788 Ki = 385 nM T52450 CM04TG 44314789 Ki = 382 nM T52450 C2BLO9 44314811 IC50 = 350 nM T52450 CSY5R3 44314812 IC50 = 430 nM T52450 C0BJ7X 44314813 IC50 = 5200 nM T52450 C7LCN0 44314824 Ki = 55000 nM T52450 CNM6W8 44314841 Ki = 193 nM T52450 C9K8JZ 44314900 Ki = 2500 nM T52450 CXRE70 44314901 Ki = 1530 nM T52450 CK3H1Y 44314929 Ki = 618 nM T52450 CS5A6Z 44314930 Ki = 296 nM T52450 CNB72W 44314931 Ki = 1050 nM T52450 CBXI30 44314932 Ki = 642 nM T52450 CCF80X 44314958 Ki = 100000 nM T52450 C3N8RQ 44314969 Ki = 10000 nM T52450 C9SRT4 44314970 Ki = 54954.09 nM T52450 C61DST 44314974 Ki = 313 nM T52450 CE2J4M 44314975 Ki = 455 nM T52450 CQE0D3 44314976 Ki = 942 nM T52450 CI2V1Y 44314995 Ki = 100000 nM T52450 C48NVD 44314999 Ki = 135 nM T52450 CB7F0J 44315000 Ki = 5000 nM T52450 CSY78M 44315028 Ki = 11200 nM T52450 CDZ5O3 44315029 Ki = 640 nM T52450 C1V9FZ 44315040 IC50 = 860 nM T52450 C02YGK 44315041 IC50 = 12000 nM T52450 C64MTA 44315075 IC50 = 630 nM T52450 C85WJB 44315076 IC50 = 1400 nM T52450 C6HW5G 44315084 Ki = 329 nM T52450 CV6KW1 44315085 Ki = 319 nM T52450 CXLD02 44315105 IC50 = 3000 nM T52450 CIJ8H3 44315114 IC50 = 2300 nM T52450 C5G7OS 44315115 IC50 = 1100 nM T52450 CBP7S0 44315139 IC50 = 970 nM T52450 C4GR1C 44315140 IC50 = 1600 nM T52450 CWS3E8 44315141 IC50 = 690 nM T52450 CPAT25 44315142 IC50 = 1600 nM T52450 C9YK1H 44315143 IC50 > 30000 nM T52450 C3VB1J 44315156 IC50 = 650 nM T52450 C79QEK 44315157 IC50 = 540 nM T52450 CAUQ47 44315167 Ki = 57543.99 nM T52450 COA01P 44315179 Ki > 50000 nM T52450 CQ1R9E 44315204 Ki = 28183.83 nM T52450 CL32FZ 44315221 Ki = 770 nM T52450 CDN4Y5 44315222 Ki = 336 nM T52450 C62FXJ 44315244 IC50 = 1100 nM T52450 CB0VI3 44315245 IC50 = 120 nM T52450 CP9M6W 44315277 Ki = 5120 nM T52450 C3SZO4 44315279 Ki = 25000 nM T52450 C4BWR2 44315286 IC50 = 22000 nM T52450 CH4YI9 44315311 IC50 = 530 nM T52450 COVF49 44315312 IC50 = 280 nM T52450 CSG05N 44315321 Ki = 313 nM T52450 COD08C 44315324 Ki = 22100 nM T52450 C50IQE 44315333 IC50 = 770 nM T52450 C1LC5H 44315334 IC50 = 1600 nM T52450 C37JMW 44315348 Ki = 39810.72 nM T52450 CKAL69 44315860 IC50 = 14 nM T52450 C0HR5Q 44316157 IC50 = 207 nM T52450 CG0JD3 44316269 Ki > 40000 nM T52450 C5RJ6F 44316310 IC50 = 597 nM T52450 CSA5P7 44316333 IC50 = 24 nM T52450 C1O6PM 44316416 Ki = 120 nM T52450 CP83EX 44316470 Ki = 37000 nM T52450 CLOS38 44316842 Ki = 90 nM T52450 CS7D5E 44317086 IC50 = 3160 nM T52450 CH70XB 44317451 IC50 = 174 nM T52450 C8Y7JG 44317981 Ki > 10000 nM T52450 C89IQW 44318090 IC50 = 3310 nM T52450 C8PLQ4 44321319 IC50 = 26 nM T52450 CT1U0G 44321321 IC50 = 44 nM T52450 C63VJF 44321390 IC50 = 183 nM T52450 C2V3KS 44321431 IC50 = 51 nM T52450 CT0O7Y 44321602 Ki = 9 nM T52450 CV8T3N 44321783 Ki = 340 nM T52450 C7Z4DQ 44321887 Ki = 36 nM T52450 CFJ20T 44321932 Ki = 53 nM T52450 C15WQO 44323336 IC50 = 45 nM T52450 C9UOW2 44323407 IC50 = 445 nM T52450 C4C1WD 44323426 IC50 = 116 nM T52450 C85JGD 44323430 IC50 = 703 nM T52450 CKP12T 44323431 IC50 = 312 nM T52450 C4R8OD 44323432 IC50 = 309 nM T52450 COQ6U7 44323456 IC50 = 91 nM T52450 CL07GT 44323526 IC50 = 618 nM T52450 CZRF63 44323527 IC50 = 690 nM T52450 CT9M4F 44323539 IC50 = 251 nM T52450 CQG24X 44323540 IC50 = 128 nM T52450 CDG29X 44324430 Ki = 31000 nM T52450 CT01XC 44324546 IC50 = 350000 nM T52450 CK5F4S 44324646 IC50 = 440000 nM T52450 C6BJ7X 44324656 IC50 = 900000 nM T52450 CT51EZ 44324668 Ki = 900 nM T52450 CV45NF 44324822 Ki = 460000 nM T52450 CCN58H 44324826 Ki = 1900000 nM T52450 CL3XT8 44324871 Ki = 18000 nM T52450 CE6VR2 44324878 IC50 = 8000000 nM T52450 CYLN13 44324879 IC50 = 10000000 nM T52450 CBI48M 44324889 IC50 = 500000 nM T52450 CEQ43S 44324934 IC50 > 10000000 nM T52450 CTOZ12 44324953 Ki = 950000 nM T52450 CO0S9J 44325072 Ki = 100 nM T52450 C4R9LM 44325085 Ki = 850 nM T52450 C21LNP 44325141 Ki = 403000 nM T52450 CL8MD0 44325156 Ki > 850 nM T52450 CV3S9G 44325157 Ki = 450 nM T52450 C9MD1A 44325159 Ki > 850 nM T52450 C6R4NI 44325225 Ki = 554 nM T52450 CRM0C1 44325233 IC50 = 258000 nM T52450 CN0GX1 44325234 IC50 = 90000 nM T52450 C5STC3 44325248 IC50 = 1600000 nM T52450 C6BRF1 44325257 Ki = 990000 nM T52450 C3M2XY 44325277 Ki = 84 nM T52450 CA4FQ5 44325443 Ki = 162 nM T52450 C20UGO 44325517 Ki > 10000 nM T52450 CHMC02 44325564 Ki = 19952.62 nM T52450 C8P6UA 44325625 Ki = 642 nM T52450 CBY75J 44325686 Ki > 10000 nM T52450 C6A1JX 44325696 Ki = 1050 nM T52450 CJU3R8 44325730 Ki = 135 nM T52450 CBV73K 44325744 Ki = 313 nM T52450 C06ZAH 44325745 Ki = 455 nM T52450 C70UFH 44325749 Ki = 319 nM T52450 C8EWP2 44325750 Ki = 313 nM T52450 C2QL0B 44325810 Ki = 382 nM T52450 CP1NU9 44325834 Ki = 942 nM T52450 C7VRX2 44325907 Ki = 193 nM T52450 C95AOR 44326036 IC50 = 121 nM T52450 CXD0V7 44326102 IC50 = 10 nM T52450 CGNU41 44326331 Ki = 224 nM T52450 CJ67MO 44326374 IC50 = 1.3 nM T52450 C3ZDL9 44326394 IC50 = 920 nM T52450 C01QWH 44326406 Ki = 3 nM T52450 CT23RH 44327170 IC50 = 20 nM T52450 C2ZH0F 44327181 IC50 = 4031 nM T52450 CC8O1F 44327205 IC50 > 10000 nM T52450 C3LBS5 44327223 IC50 = 4600 nM T52450 CCY3J1 44327232 IC50 = 30 nM T52450 C0WX4Z 44327233 IC50 > 10000 nM T52450 CP5B1W 44327235 IC50 = 1500 nM T52450 CVR1S3 44327236 IC50 = 1900 nM T52450 CP79CH 44327243 IC50 > 10000 nM T52450 CC8IX0 44327244 IC50 > 1000 nM T52450 CJF81U 44327375 IC50 > 10000 nM T52450 C8V3AO 44327386 IC50 = 870.96 nM T52450 CDL26B 44327405 IC50 = 7000 nM T52450 C0UC5H 44327407 IC50 = 2951.21 nM T52450 C6TPB1 44327409 IC50 = 476 nM T52450 CRPT39 44327418 IC50 > 10000 nM T52450 C2V1BQ 44327419 IC50 > 10000 nM T52450 C12NGR 44327430 IC50 = 4100 nM T52450 CM2E3F 44327431 IC50 > 10000 nM T52450 C8ZI0P 44327432 IC50 = 10000 nM T52450 CVJ9Q6 44327443 IC50 = 331.13 nM T52450 C4R9WM 44327681 IC50 = 927 nM T52450 CR40TV 44327695 IC50 > 10000 nM T52450 C6IM7G 44327755 IC50 = 1905.46 nM T52450 C85QTP 44328155 IC50 = 70000 nM T52450 CZQ6N7 44328189 IC50 = 50000 nM T52450 CDC32P 44328337 IC50 = 2120 nM T52450 C8C1HG 44328339 IC50 = 1630 nM T52450 CKLD96 44328378 IC50 = 730 nM T52450 C2B3WH 44328379 IC50 = 150 nM T52450 CX5H2A 44328380 IC50 = 360 nM T52450 C1NST6 44328467 IC50 = 190 nM T52450 C86QAY 44328559 IC50 = 37000 nM T52450 CHU2P7 44328876 IC50 = 24 nM T52450 C0KA4S 44328937 IC50 = 171 nM T52450 CLT8B6 44328971 IC50 = 35 nM T52450 C7J0ZI 44329016 IC50 = 763 nM T52450 CMLA39 44329018 IC50 = 18 nM T52450 CW24VN 44329040 IC50 = 59 nM T52450 C9J0VO 44329253 IC50 = 61 nM T52450 C90CHA 44329405 IC50 = 30 nM T52450 C2PB4Z 44329622 IC50 = 800 nM T52450 CI3Z4K 44329623 IC50 = 6 nM T52450 C6OL8M 44329636 IC50 = 60 nM T52450 CB0G1H 44329644 IC50 = 1000 nM T52450 CA65RO 44329672 IC50 = 50 nM T52450 CK9HO7 44329673 IC50 = 20 nM T52450 C07GRS 44329693 IC50 = 10 nM T52450 CBH16R 44329694 IC50 = 6 nM T52450 CG3E7A 44329712 IC50 = 2 nM T52450 C9SN6I 44329713 IC50 = 30 nM T52450 CZ2FW6 44329725 IC50 = 10 nM T52450 CDKI48 44329741 IC50 = 9 nM T52450 CK3M2H 44329742 IC50 = 20 nM T52450 C39RDS 44329886 IC50 = 6 nM T52450 C63RHP 44329909 IC50 = 10 nM T52450 CVQA75 44329910 IC50 = 5 nM T52450 C84SLI 44329926 IC50 = 9 nM T52450 CJS6B1 44329927 IC50 = 5 nM T52450 C2K6OU 44329943 IC50 > 1000 nM T52450 C5BYR4 44329998 IC50 > 10000 nM T52450 C0SMC9 44330092 IC50 = 26 nM T52450 C35SIO 44330094 IC50 = 140 nM T52450 C3NM2G 44330095 IC50 = 6.761 nM T52450 C6SCU5 44330119 IC50 = 2.3 nM T52450 C69KPL 44330130 IC50 = 2300 nM T52450 C9P6ZF 44330131 IC50 = 229.09 nM T52450 CKS01F 44330133 IC50 > 10000 nM T52450 C1IE0S 44330147 IC50 > 100000 nM T52450 CXI49L 44330197 IC50 > 10000 nM T52450 CDQM84 44330198 IC50 = 5.7 nM T52450 CH6EN4 44330225 IC50 > 10000 nM T52450 C3GA9Q 44330226 IC50 = 28 nM T52450 CD0L6S 44331932 IC50 = 444 nM T52450 CHIG68 44331976 IC50 = 129 nM T52450 CF4JN0 44331983 IC50 = 343 nM T52450 CG2AH4 44331984 IC50 = 745 nM T52450 CPB96A 44332003 IC50 = 517 nM T52450 C6RE3I 44332107 IC50 = 82 nM T52450 C3L1HQ 44332161 IC50 = 674 nM T52450 CG2Q8W 44332306 IC50 > 1000 nM T52450 CY0MQ9 44332313 IC50 = 150 nM T52450 CR4PF3 44333557 IC50 = 270 nM T52450 C4IBF6 44333558 IC50 = 330 nM T52450 CPI95O 44333573 IC50 = 17 nM T52450 CW97JB 44333575 IC50 = 220 nM T52450 CCZ57P 44333576 IC50 = 340 nM T52450 CZB5U7 44333614 IC50 = 230 nM T52450 C2RO8K 44333616 IC50 = 320 nM T52450 CXO36Z 44333646 IC50 = 140 nM T52450 CPJ92E 44333652 IC50 > 100000 nM T52450 CF2L8K 44333653 IC50 = 290 nM T52450 CW2RF9 44333861 IC50 > 100000 nM T52450 C8U7ZO 44334049 IC50 = 160 nM T52450 CFP3X8 44334949 IC50 = 384 nM T52450 CV5RF0 44334963 IC50 = 25170 nM T52450 C4AOZ7 44334981 IC50 = 8760 nM T52450 CXW59C 44334982 IC50 = 458 nM T52450 CCH1W8 44334983 IC50 = 117 nM T52450 CQ0UI1 44335017 IC50 = 1620 nM T52450 CX58SB 44335240 IC50 = 198 nM T52450 CA96JG 44335285 IC50 = 654 nM T52450 CM3F2G 44337397 IC50 > 10000 nM T52450 CE70RM 44337427 IC50 > 10000 nM T52450 CDW4I0 44337430 IC50 = 500 nM T52450 C8GR3H 44337445 IC50 > 10000 nM T52450 CJ6MP1 44337450 IC50 < 100 nM T52450 C9L3HU 44337570 IC50 = 5000 nM T52450 C5ONP9 44337593 IC50 > 10000 nM T52450 CD5ZE7 44337599 IC50 > 1000 nM T52450 C0Y2CZ 44339375 IC50 = 830 nM T52450 CP12TJ 44339394 IC50 = 1300 nM T52450 COR15M 44339402 IC50 = 12000 nM T52450 CU5NI2 44339444 IC50 = 1500 nM T52450 CISO73 44339448 IC50 = 3400 nM T52450 C4QKI6 44339451 IC50 = 19 nM T52450 CEUP59 44339452 IC50 = 1400 nM T52450 CU7DZ9 44339462 IC50 = 6400 nM T52450 CI5X0G 44339523 IC50 = 1.9 nM T52450 CB9K8T 44339536 IC50 = 13 nM T52450 CLT8C6 44339543 IC50 = 1700 nM T52450 C6M4UR 44339544 IC50 = 10000 nM T52450 C2CRY1 44339556 IC50 = 14 nM T52450 CTBU53 44339564 IC50 = 4.7 nM T52450 C58OSK 44339567 IC50 = 2.7 nM T52450 C5PQ1B 44339569 IC50 = 1900 nM T52450 CA65PF 44339570 IC50 = 3800 nM T52450 C4W8LS 44339571 IC50 = 12000 nM T52450 CX2KJ3 44339574 IC50 = 180 nM T52450 COUE24 44339575 IC50 = 6700 nM T52450 CEK3G0 44339588 IC50 = 60 nM T52450 C0WP9C 44339590 IC50 = 6.2 nM T52450 CE90PW 44339624 IC50 = 17000 nM T52450 CMA2L3 44339647 IC50 = 1500 nM T52450 CFCZ60 44339648 IC50 = 2200 nM T52450 C5C2LI 44339654 IC50 = 5.1 nM T52450 CH3I5B 44339870 Ki >= 10000 nM T52450 CM6VJ2 44339884 Ki >= 10000 nM T52450 CMVE19 44339885 Ki >= 10000 nM T52450 CLD2P9 44339900 Ki >= 10000 nM T52450 C5R6KD 44339905 Ki >= 10000 nM T52450 C3B5XK 44339917 Ki >= 10000 nM T52450 C2D6VN 44339918 Ki >= 10000 nM T52450 CRQJ09 44339936 Ki >= 10000 nM T52450 C07CVA 44340076 IC50 = 30000 nM T52450 C4JLG8 44340091 Ki >= 10000 nM T52450 CLKT58 44340092 Ki >= 10000 nM T52450 C4KLU8 44340093 Ki >= 10000 nM T52450 CXW34P 44340094 Ki >= 10000 nM T52450 CZ45CH 44340125 IC50 = 50 nM T52450 CZ98KU 44340156 Ki >= 10000 nM T52450 C7E5FI 44340159 Ki >= 10000 nM T52450 CGV94P 44340160 Ki >= 10000 nM T52450 C3IS1O 44340161 Ki >= 10000 nM T52450 CPK5W0 44340172 Ki >= 10000 nM T52450 C4SC6L 44340175 IC50 > 32000 nM T52450 CVJM53 44340176 IC50 = 4100 nM T52450 CDR5V6 44340199 Ki >= 10000 nM T52450 C7PAI6 44340200 Ki >= 10000 nM T52450 CJ4Z9W 44340207 Ki >= 10000 nM T52450 CZ31VY 44340208 Ki >= 10000 nM T52450 CVG1R5 44340217 Ki >= 10000 nM T52450 C39EMX 44340229 Ki >= 10000 nM T52450 C4B9QZ 44340327 Ki >= 10000 nM T52450 C2XY8H 44340328 Ki >= 10000 nM T52450 CUM9J0 44340329 Ki >= 10000 nM T52450 CAT48Z 44340657 Ki = 2090 nM T52450 CJBC96 44340662 Ki = 72 nM T52450 CJ83VB 44340663 Ki = 13000 nM T52450 C3CYZ8 44340673 Ki = 1800 nM T52450 CRI8Q4 44340696 Ki = 6800 nM T52450 CF1QZ3 44340718 Ki = 7200 nM T52450 C09ILT 44340727 Ki = 5800 nM T52450 C6AS8J 44340740 Ki = 3400 nM T52450 CAC07H 44340742 Ki = 1790 nM T52450 CPVL28 44340743 Ki = 1090 nM T52450 CH8BO5 44340744 Ki = 1100 nM T52450 CQ4RT5 44340809 Ki = 3330 nM T52450 CL0U9T 44340810 Ki = 870 nM T52450 CV6W7Z 44340812 Ki = 4410 nM T52450 CW53EF 44340868 Ki = 5810 nM T52450 C6ZDV3 44340869 Ki = 3890 nM T52450 CR1ID4 44340923 Ki = 1600 nM T52450 CL9I4M 44341538 Ki = 1087 nM T52450 CT82PD 44341747 IC50 <= 100 nM T52450 C0GC5F 44341759 IC50 = 25 nM T52450 CE0PL2 44341937 IC50 = 550 nM T52450 C83FUZ 44341941 IC50 = 31 nM T52450 C2S1GO 44341947 IC50 = 750 nM T52450 C5S0YH 44341969 IC50 = 21 nM T52450 C5FG4N 44341974 IC50 = 5900 nM T52450 CN4UP5 44341977 IC50 = 3800 nM T52450 C2S7PL 44341987 IC50 = 330 nM T52450 C6EY7C 44342019 IC50 = 8800 nM T52450 CK4WL8 44342020 IC50 = 9600 nM T52450 C8WH0C 44342056 IC50 = 870 nM T52450 CT68XS 44342103 IC50 = 12000 nM T52450 C8LG0S 44342114 IC50 = 8 nM T52450 CWYV36 44342115 IC50 = 1700 nM T52450 CER9M5 44342120 IC50 = 500 nM T52450 C0KO4U 44342125 IC50 = 780 nM T52450 CD59OJ 44342127 IC50 = 42 nM T52450 CA1X5L 44342131 IC50 = 550 nM T52450 CIS5M3 44342135 IC50 = 3900 nM T52450 C80EKJ 44342143 IC50 = 3900 nM T52450 C29IPJ 44342160 IC50 = 1200 nM T52450 C8MFA9 44342168 IC50 = 930 nM T52450 CXWQ20 44342181 IC50 = 1250 nM T52450 CVNF08 44342224 IC50 = 1400 nM T52450 CN9J4G 44342228 IC50 = 3000 nM T52450 C5PAS4 44342236 IC50 = 4900 nM T52450 CE1TJ7 44342237 IC50 > 10000 nM T52450 CMI0T2 44342251 IC50 = 4800 nM T52450 CC1JA5 44342253 IC50 = 106 nM T52450 CAN54Y 44342308 IC50 = 550 nM T52450 CURT86 44342353 Ki > 30000 nM T52450 CR9G4Y 44342410 IC50 = 110 nM T52450 CT3EL5 44342419 IC50 = 1900 nM T52450 CD3Y9N 44342428 IC50 = 180 nM T52450 CG0X7W 44342441 IC50 > 10000 nM T52450 CSJL84 44342528 Ki = 4 nM T52450 C6Y8JA 44342529 Ki = 4 nM T52450 CNP86Q 44342537 Ki = 3 nM T52450 C4TSH9 44342583 Ki = 2 nM T52450 C2SZB1 44342614 IC50 = 5 nM T52450 CT28SZ 44342640 Ki = 3 nM T52450 CV3AD2 44342666 Ki = 5 nM T52450 C0P1ZX 44342686 Ki = 2 nM T52450 C8PMR6 44342688 Ki = 5 nM T52450 CMPF49 44342715 Ki = 1 nM T52450 CZR09J 44342848 Ki = 2 nM T52450 C0U9NM 44342916 Ki = 6 nM T52450 C51RKI 44342965 Ki = 1 nM T52450 C2SD0P 44342985 Ki = 3 nM T52450 CT6UP7 44342986 Ki = 12 nM T52450 C8G7WL 44344564 Ki = 300 nM T52450 CD43AB 44344565 Ki = 180 nM T52450 CBH9I5 44344658 IC50 = 5900 nM T52450 CC29QO 44344739 Ki > 100 nM T52450 CWA42F 44344746 Ki = 1400 nM T52450 CQPN17 44344749 Ki = 8400 nM T52450 CL41FG 44344753 Ki = 8500 nM T52450 C3V0GM 44348957 IC50 = 29 nM T52450 CFI6N5 44348963 IC50 = 47 nM T52450 CCF94Z 44349787 IC50 = 70000 nM T52450 C1L2GF 44350073 IC50 = 4400 nM T52450 CQ5RN6 44350101 IC50 = 6600 nM T52450 CE2X3Q 44350116 IC50 > 100000 nM T52450 CCHG20 44352499 IC50 = 980 nM T52450 C78IPJ 44352500 IC50 = 3 nM T52450 CK4O5E 44352718 IC50 = 22 nM T52450 CO9R4W 44356376 Ki > 4949 nM T52450 C3MZA1 44356386 Ki > 4949 nM T52450 CH1E2S 44356406 Ki > 4949 nM T52450 C84LUM 44356631 Ki > 4949 nM T52450 CG6T9A 44356632 Ki > 4949 nM T52450 C3WFH7 44356634 Ki > 4949 nM T52450 CB8KY4 44356635 Ki > 4949 nM T52450 COIA82 44356636 Ki > 4949 nM T52450 C4BU6T 44356644 Ki > 4949 nM T52450 CH9YT4 44356659 Ki > 4949 nM T52450 CD96OP 44356667 IC50 > 100000 nM T52450 C83BTI 44356670 Ki = 510 nM T52450 CH4V6J 44356671 Ki = 850 nM T52450 C68LMR 44356675 Ki > 4949 nM T52450 C69YIP 44356686 Ki > 4949 nM T52450 CT05XN 44356687 Ki > 4949 nM T52450 CO5XG6 44356688 IC50 > 60000 nM T52450 CML03W 44356689 Ki > 4949 nM T52450 CQ4NP5 44356690 Ki > 4949 nM T52450 CZQF75 44356702 IC50 = 10600 nM T52450 C1A4NY 44356703 IC50 = 500 nM T52450 CE8U2Y 44356714 Ki > 4949 nM T52450 C4NM2V 44356737 Ki = 1200 nM T52450 CE81GS 44356767 IC50 > 60000 nM T52450 C0BRH3 44356774 IC50 > 60000 nM T52450 C4G3KR 44356775 IC50 > 60000 nM T52450 C9DIQ5 44356789 IC50 = 2000 nM T52450 CO3RI0 44356790 IC50 = 23900 nM T52450 C8XA0M 44356791 IC50 = 7500 nM T52450 CCY5U3 44356804 IC50 = 61 nM T52450 C25ZQU 44356805 IC50 = 52100 nM T52450 C27LMU 44356852 Ki > 4949 nM T52450 CTU64D 44356889 Ki > 4949 nM T52450 C4TM1I 44356890 Ki > 4949 nM T52450 C1WA4B 44356906 Ki > 4949 nM T52450 C50ELY 44356907 Ki > 4949 nM T52450 CVU8L2 44356924 Ki > 4949 nM T52450 CD1GW2 44356953 Ki > 4949 nM T52450 C1YAR5 44356962 Ki = 1100 nM T52450 C2Y4KQ 44356963 Ki > 10000 nM T52450 CJH1C3 44356964 Ki = 1000 nM T52450 CR41QN 44356969 Ki > 4949 nM T52450 C3BT0N 44356971 Ki > 4949 nM T52450 C81OIZ 44356983 Ki > 4949 nM T52450 CHNC03 44356993 Ki > 4949 nM T52450 C9Z3RT 44356998 Ki > 4949 nM T52450 CR4A7G 44356999 Ki > 4949 nM T52450 C2VS6P 44357000 Ki > 4949 nM T52450 CEI0X5 44357004 IC50 = 17800 nM T52450 CES1G8 44357007 Ki > 4949 nM T52450 C6NQ7K 44357012 Ki > 4949 nM T52450 C2HIN3 44357023 Ki > 4949 nM T52450 CI4JO7 44357024 Ki > 4949 nM T52450 CW4VQ3 44357029 Ki > 4949 nM T52450 C2AIT6 44357209 Ki > 4949 nM T52450 CJK2P7 44357220 Ki > 4949 nM T52450 CIX6G5 44357225 Ki > 4949 nM T52450 CQ60YD 44360219 IC50 = 61 nM T52450 CT4C6P 44360260 IC50 = 217 nM T52450 CY5I3O 44360286 IC50 = 22 nM T52450 C40OCB 44360287 IC50 = 1 nM T52450 C3IW9L 44360784 IC50 = 2.4 nM T52450 CH72OI 44363783 IC50 = 730 nM T52450 CGQ92A 44364037 IC50 = 462 nM T52450 C36YLM 44364111 IC50 = 13190 nM T52450 CN4T7Q 44364119 IC50 = 0.041 nM T52450 CH4TE7 44364121 IC50 = 452 nM T52450 CPE91Y 44364122 IC50 = 152 nM T52450 CG2X0C 44364224 IC50 = 6319 nM T52450 C1F8XN 44364249 IC50 = 123 nM T52450 CWM47H 44364250 IC50 = 595 nM T52450 CJ2B8F 44364280 IC50 = 15020 nM T52450 C90CYD 44367175 IC50 = 255 nM T52450 C2DV0R 44367276 IC50 = 74 nM T52450 C5BAW2 44367284 IC50 = 86 nM T52450 C2YG5E 44367285 IC50 = 4235 nM T52450 CUDF82 44367309 IC50 = 790 nM T52450 C92OKS 44369679 Ki > 850 nM T52450 C63WRQ 44369680 Ki = 13.2 nM T52450 CHV7Z8 44369681 Ki = 10.5 nM T52450 CX4ZU6 44369702 Ki = 31.4 nM T52450 C8ZK2I 44369876 Ki > 850 nM T52450 C1QWA3 44374051 IC50 = 19 nM T52450 CX01WF 44374220 IC50 = 44 nM T52450 C40TSF 44374235 IC50 = 74 nM T52450 C1I6QU 44374342 IC50 = 103 nM T52450 CZYL14 44374353 IC50 = 51 nM T52450 CGK04Y 44374370 IC50 = 211 nM T52450 CCZ6J3 44379232 Ki = 4620 nM T52450 CW20ML 44379249 Ki = 1600 nM T52450 CXM06G 44379250 Ki > 10000 nM T52450 CK0B1D 44379273 Ki > 10000 nM T52450 COD6P1 44379499 Ki > 10000 nM T52450 C84YPO 44379547 Ki > 10000 nM T52450 C4M3CU 44380421 Ki = 15 nM T52450 C0CH2Q 44380422 Ki = 13 nM T52450 CBLY46 44380446 Ki = 33 nM T52450 C0F6ZP 44380458 Ki = 85 nM T52450 C1VY9Q 44380628 Ki = 72 nM T52450 C4H8SW 44380647 Ki = 198 nM T52450 CY03NT 44380706 Ki = 18 nM T52450 CJ5W2S 44381004 Ki = 282 nM T52450 C82UHB 44381005 Ki = 25 nM T52450 C8A9FK 44381033 Ki = 0.6 nM T52450 C3LIF2 44381197 Ki = 53 nM T52450 C27DGC 44381207 Ki = 16 nM T52450 C70VDN 44381208 Ki = 22 nM T52450 CMCN65 44383696 IC50 = 525 nM T52450 CYE90S 44383704 Ki = 10.7 nM T52450 C4O9DP 44383747 Ki = 1.81 nM T52450 C0W2SV 44383786 Ki = 6.5 nM T52450 C2UNW6 44383789 Ki = 3.64 nM T52450 C6V9FQ 44383801 Ki = 4.43 nM T52450 CV8UX5 44383829 Ki = 39.8 nM T52450 CCY30B 44383847 Ki = 7.33 nM T52450 C7MLD8 44383849 Ki = 6.67 nM T52450 C9F5LS 44384003 Ki = 18.7 nM T52450 CSM3P7 44384004 Ki = 58.8 nM T52450 CO9LJ6 44384005 Ki = 17.4 nM T52450 CJ4NV9 44384173 Ki = 24 nM T52450 C7B3AN 44384343 Ki = 10.7 nM T52450 C4B9NU 44384357 Ki = 27.1 nM T52450 CC81JP 44384395 Ki = 2.02 nM T52450 CKG95Y 44384455 Ki > 850 nM T52450 C96PAY 44384542 Ki = 3.14 nM T52450 C7HA0F 44384590 Ki = 0.97 nM T52450 C5ZYN1 44384591 Ki = 4.9 nM T52450 CVZ42A 44384592 Ki = 160 nM T52450 CSV63O 44384594 IC50 = 608 nM T52450 C49TAV 44384649 Ki = 11.4 nM T52450 CALI01 44384650 Ki = 6.75 nM T52450 C7A2HC 44384755 Ki = 20.1 nM T52450 CL51XE 44384756 Ki = 4.1 nM T52450 CD2PM4 44384761 Ki = 9.65 nM T52450 CJH8P4 44384762 Ki > 850 nM T52450 CH3M5X 44384813 Ki = 17.8 nM T52450 C59NBH 44384814 Ki = 10.9 nM T52450 C3EV2A 44384940 IC50 > 2000 nM T52450 C0XE8K 44384941 IC50 > 2000 nM T52450 C5AE0O 44384972 Ki = 20.8 nM T52450 C3IJO9 44384994 IC50 > 2000 nM T52450 CK7RP9 44385344 Ki = 5.39 nM T52450 CZ5I8B 44386229 IC50 > 10000 nM T52450 C1FMN0 44386697 IC50 = 1100 nM T52450 CZ6PU7 44389401 Ki > 5000 nM T52450 CO4W0Y 44389552 Ki > 5000 nM T52450 C3YPG6 44390245 IC50 = 114 nM T52450 CAC3F2 44390281 IC50 = 576 nM T52450 CRE9G2 44390289 IC50 = 171 nM T52450 CN41JE 44390299 IC50 = 207 nM T52450 C5VBL2 44390300 IC50 = 142 nM T52450 C47EZV 44390314 IC50 = 4584 nM T52450 CF65OK 44390317 IC50 = 277 nM T52450 C3GU1Q 44390323 IC50 = 212 nM T52450 CAZ2B4 44390326 IC50 = 3031 nM T52450 CYW89M 44390352 IC50 = 1136 nM T52450 CPK9Z6 44390355 IC50 = 334 nM T52450 CEJH75 44390356 IC50 = 285 nM T52450 CWYM93 44390391 IC50 = 645 nM T52450 CC7QW9 44391352 IC50 = 13000 nM T52450 CMGB67 44393214 IC50 = 356 nM T52450 CA1S5T 44393217 IC50 = 852 nM T52450 CBO9E6 44393239 IC50 = 1255 nM T52450 CT1LM8 44393266 IC50 = 682 nM T52450 C0SGF6 44393279 IC50 = 483 nM T52450 CYFC07 44393295 IC50 = 904 nM T52450 C24INM 44393328 IC50 = 456 nM T52450 C15IZJ 44393358 IC50 = 578 nM T52450 C3HP5Q 44393383 IC50 = 238 nM T52450 CS06PD 44393394 IC50 = 813 nM T52450 CFA83O 44393414 IC50 = 853 nM T52450 C89FTQ 44393434 Ki > 4900 nM T52450 CCO3S9 44393444 Ki > 4900 nM T52450 CNO4P6 44393516 Ki > 4900 nM T52450 C5OIK4 44393520 Ki > 4900 nM T52450 CDG2K7 44393747 IC50 = 120 nM T52450 CWUV21 44393760 IC50 = 10000 nM T52450 CQ6WZ5 44393836 IC50 = 22000 nM T52450 CR58XA 44393837 IC50 = 5400 nM T52450 CIH8T9 44393838 IC50 > 30000 nM T52450 CFR4G2 44393892 IC50 < 30 nM T52450 CMBJ97 44393897 IC50 < 3 nM T52450 CF3M5K 44393910 IC50 = 27000 nM T52450 C4YJI9 44393913 IC50 > 30000 nM T52450 C0E8BQ 44393936 IC50 = 19000 nM T52450 CGU63Q 44393964 IC50 > 30000 nM T52450 C8P0IG 44393980 IC50 = 13000 nM T52450 CP24NE 44394027 IC50 = 4700 nM T52450 CHP81Z 44394038 IC50 = 270 nM T52450 CKB7S1 44394067 IC50 > 30000 nM T52450 C80NZE 44394179 Ki > 4900 nM T52450 CBDW36 44394383 IC50 = 500 nM T52450 C7SI6E 44394425 IC50 = 1100 nM T52450 CN7WS6 44394426 IC50 = 420 nM T52450 C1TWP6 44394594 Ki > 100000 nM T52450 CG01SR 44394595 Ki > 200000 nM T52450 CV6YR1 44394601 Ki > 300000 nM T52450 C6OM9B 44394637 Ki = 92000 nM T52450 CZ05UP 44394668 Ki > 200000 nM T52450 CAFL18 44394671 Ki = 30000 nM T52450 CGQ98X 44394681 Ki = 32000 nM T52450 CQM90E 44394682 Ki = 46000 nM T52450 C8MY4S 44394703 Ki > 100000 nM T52450 CGS56H 44394744 Ki > 100000 nM T52450 CFBA04 44394754 Ki > 100000 nM T52450 CK5X6F 44394758 Ki > 400000 nM T52450 C3TQS0 44394797 Ki = 64000 nM T52450 CN6GO3 44394819 IC50 = 340 nM T52450 C79OYF 44394821 Ki > 300000 nM T52450 CVGU01 44394916 IC50 = 270 nM T52450 CG1W0V 44394994 IC50 = 180 nM T52450 CT6VX4 44395030 IC50 = 860 nM T52450 C2EG4V 44395069 IC50 = 2600 nM T52450 CT5N1F 44395157 IC50 = 310 nM T52450 CSMF27 44395269 IC50 = 2700 nM T52450 CBG4Q5 44395271 IC50 = 600 nM T52450 CGKI40 44395434 IC50 = 1300 nM T52450 C3Z6DG 44395454 IC50 = 1600 nM T52450 CZB81D 44395506 IC50 = 310 nM T52450 CPJ4G7 44395643 IC50 = 190 nM T52450 CC05MG 44395660 IC50 = 120 nM T52450 CNQ6C0 44395935 IC50 = 120 nM T52450 C3UO7Y 44395976 IC50 = 7800 nM T52450 CAV7Z6 44396001 IC50 = 520 nM T52450 CTDR73 44396048 IC50 = 1600 nM T52450 CKV57D 44399071 IC50 = 773 nM T52450 C0NSO4 44399233 IC50 = 5100 nM T52450 CRL5D0 44399252 IC50 = 690 nM T52450 CHL9S2 44399294 Ki > 4950 nM T52450 CD49UI 44399312 Ki > 4950 nM T52450 C7IDB0 44399341 IC50 = 255 nM T52450 C2UDW8 44399397 IC50 = 170 nM T52450 CA0DV5 44399432 IC50 = 198 nM T52450 C95RKA 44399451 IC50 = 2300 nM T52450 CIA8T3 44399555 Ki > 4950 nM T52450 CV2CQ0 44399635 IC50 = 790 nM T52450 CJWB10 44399637 IC50 = 1100 nM T52450 CW83LM 44399638 IC50 = 592 nM T52450 C7XCI6 44399665 IC50 = 290 nM T52450 CW9MD1 44399704 IC50 = 1500 nM T52450 C2JMC1 44399712 IC50 = 679 nM T52450 CD8Q2Y 44399731 IC50 = 715 nM T52450 CC16YQ 44399733 IC50 = 100 nM T52450 C91POV 44402021 IC50 = 10000 nM T52450 CYCJ78 44402280 IC50 = 397 nM T52450 CD2X7N 44404429 IC50 = 121 nM T52450 C3I8NA 44404458 IC50 = 121 nM T52450 CIXM04 44404472 IC50 = 121 nM T52450 C01XOM 44404480 Ki = 3 nM T52450 C7DI5L 44404488 Ki = 3 nM T52450 CZ3NO9 44404495 IC50 = 1.3 nM T52450 CY6WL5 44404502 IC50 = 34000 nM T52450 CWGQ46 44404503 IC50 = 37100 nM T52450 CLXM58 44404504 IC50 = 28000 nM T52450 CYE6A7 44404505 IC50 = 1.3 nM T52450 CTP76G 44404512 IC50 = 121 nM T52450 C9LAQ1 44404514 Ki = 3 nM T52450 CY6E1J 44404533 IC50 = 1.3 nM T52450 CIT3P8 44404534 IC50 = 920 nM T52450 C9DNC1 44404535 Ki = 3 nM T52450 C9EC1T 44404536 IC50 = 3 nM T52450 CN1O3X 44404539 Ki = 70 nM T52450 CO4G0A 44404541 Ki = 70 nM T52450 CBJ13Q 44404548 Ki = 8.2 nM T52450 CFY29O 44404552 Ki = 70 nM T52450 C30DKN 44404553 IC50 = 22 nM T52450 CJHP37 44404556 Ki = 8.2 nM T52450 CJ26OA 44404557 IC50 = 22 nM T52450 CE3TB5 44404559 Ki = 70 nM T52450 C0O9PC 44404565 Ki = 8.2 nM T52450 CCV50A 44404569 Ki = 8.2 nM T52450 C14OTW 44404579 Ki = 224 nM T52450 C30YXK 44404585 IC50 = 10 nM T52450 CX5UQ3 44404587 Ki = 224 nM T52450 CU7F9R 44404610 IC50 = 10 nM T52450 C2P9ED 44404613 Ki = 224 nM T52450 C3Y0VU 44404620 IC50 = 10 nM T52450 CC3E9A 44404625 Ki = 224 nM T52450 C4L8NX 44404630 IC50 = 10 nM T52450 C7Z0OH 44404761 IC50 = 1248 nM T52450 CIC60V 44406452 IC50 > 100000 nM T52450 C1F0DR 44406571 IC50 > 10000 nM T52450 CHM26J 44406652 Ki = 2500 nM T52450 C1K3QM 44406655 IC50 = 30 nM T52450 C6YG5S 44406678 IC50 > 1000 nM T52450 CT7CD3 44409041 IC50 = 35 nM T52450 CJ2Q8Z 44409042 IC50 = 159 nM T52450 CY3KF2 44409047 IC50 = 101 nM T52450 CT01JW 44409066 IC50 = 26 nM T52450 CJNE37 44409163 IC50 = 42 nM T52450 CVA69I 44409164 IC50 = 87 nM T52450 C9I0JW 44409184 IC50 = 1052 nM T52450 C1JSU2 44409197 IC50 = 300 nM T52450 CW4BM3 44409214 IC50 = 11 nM T52450 CVRL76 44409215 IC50 = 7 nM T52450 C9F7HR 44409221 IC50 = 7 nM T52450 CJ70LK 44409222 IC50 = 29 nM T52450 C5J1PS 44409261 IC50 = 2 nM T52450 C06EZF 44409365 IC50 = 17 nM T52450 CV5AW8 44409366 IC50 = 35 nM T52450 C9PS4Q 44409369 IC50 = 21 nM T52450 C1S4GD 44409389 IC50 = 19 nM T52450 C69CGM 44409390 IC50 = 21 nM T52450 C1SKI7 44409405 IC50 = 33 nM T52450 C84ZSL 44411052 Ki = 0.7 nM T52450 CUE29K 44411053 Ki = 83 nM T52450 C6IKL1 44411602 IC50 > 1000 nM T52450 CEB0S4 44411823 IC50 > 1000 nM T52450 CVM7Y3 44413975 IC50 = 4150 nM T52450 C4X0GA 44413977 IC50 = 1850 nM T52450 CH01EO 44413978 IC50 = 4700 nM T52450 CQ8HK9 44413979 IC50 = 5460 nM T52450 CBT0P2 44413982 IC50 = 3010 nM T52450 C9BA0V 44413987 IC50 = 6980 nM T52450 CDUI73 44413992 IC50 = 65 nM T52450 CHN85S 44414002 IC50 = 6600 nM T52450 C2OJ4B 44414029 IC50 = 7970 nM T52450 CZ5KM8 44421257 IC50 > 10000 nM T52450 CT5PC9 44422672 IC50 = 98 nM T52450 CS9D5U 44422720 IC50 = 450 nM T52450 CNWM05 44422723 IC50 = 600 nM T52450 C58LAY 44422724 IC50 = 160 nM T52450 CDQU41 44422736 IC50 = 590 nM T52450 CVUB56 44422737 IC50 = 320 nM T52450 CB8G2W 44422743 IC50 = 320 nM T52450 CO24JF 44423677 IC50 = 110000 nM T52450 C8BHL5 44431844 IC50 > 5000 nM T52450 CR1DN9 44431845 IC50 > 5000 nM T52450 CHFB16 44431846 IC50 > 5000 nM T52450 C0C3ZT 44431847 IC50 > 5000 nM T52450 CS49GV 44431848 IC50 > 5000 nM T52450 C4AVK5 44431849 IC50 > 5000 nM T52450 C5DH4Q 44431850 IC50 > 5000 nM T52450 CLHE45 44431851 IC50 > 5000 nM T52450 CYG29L 44431852 IC50 > 5000 nM T52450 C4OF5L 44431853 IC50 > 5000 nM T52450 CWU7G8 44434565 IC50 = 32000 nM T52450 CF9HU5 44434566 IC50 = 9130 nM T52450 CV3M6F 44434578 IC50 = 1240 nM T52450 C70MGQ 44440455 Ki > 4946 nM T52450 CDY53F 44440460 Ki > 4946 nM T52450 CTB9P6 44440461 Ki = 988 nM T52450 C63RLK 44440462 Ki > 4946 nM T52450 C23JBO 44440463 Ki > 4946 nM T52450 CT9P3Y 44440464 Ki > 4946 nM T52450 CX32AM 44440465 Ki > 4946 nM T52450 C6FOC7 44440466 Ki > 4946 nM T52450 CMPX37 44440467 Ki > 4946 nM T52450 CV4F6Z 44440468 Ki > 4946 nM T52450 C6K8VB 44440469 Ki > 4946 nM T52450 C4Y0UM 44440470 Ki > 4946 nM T52450 CHU49A 44440471 Ki > 4946 nM T52450 C0HX1L 44445199 IC50 = 31000 nM T52450 CPQT35 44445200 IC50 = 25000 nM T52450 C2X6IP 44445201 IC50 = 37000 nM T52450 CSRB79 44445202 IC50 = 50000 nM T52450 C2O6KZ 44445203 IC50 = 32000 nM T52450 CASF34 44445204 IC50 = 30000 nM T52450 CQZ6M0 44445205 IC50 = 47000 nM T52450 CH7Z5M 44445206 IC50 = 65000 nM T52450 C71CPO 44445207 IC50 = 28000 nM T52450 CO9QA4 44445209 IC50 = 69000 nM T52450 CH3UQ5 44445210 IC50 = 99000 nM T52450 C6B4LG 44445211 IC50 = 59000 nM T52450 C1WA5N 44445212 IC50 = 67000 nM T52450 CM2CD0 44445213 IC50 = 64000 nM T52450 C6ZX2P 44445214 IC50 = 28000 nM T52450 C9KE8P 44445215 IC50 = 23000 nM T52450 C68QEF 44445216 IC50 = 35000 nM T52450 CCK7W2 44445217 IC50 = 70000 nM T52450 C58BQA 44445218 IC50 = 41000 nM T52450 C4CGN2 44445219 IC50 = 16000 nM T52450 C1IVR6 44445220 IC50 = 30000 nM T52450 CG2U7H 44445221 IC50 = 19000 nM T52450 CVW48J 44445222 IC50 = 51000 nM T52450 CL3HZ8 44445223 IC50 = 26000 nM T52450 CPY73U 44445224 IC50 = 19000 nM T52450 C9MA2F 44445225 IC50 = 22000 nM T52450 C9SJM3 44445226 IC50 = 81000 nM T52450 CH91WG 44445228 IC50 = 86000 nM T52450 CO59HI 44445229 IC50 = 115000 nM T52450 C62WPE 44445230 IC50 = 75000 nM T52450 COIR35 44445231 IC50 = 128000 nM T52450 CBH0M7 44445233 IC50 = 42000 nM T52450 CIS7M5 44445234 IC50 = 68000 nM T52450 CKN60A 44445235 IC50 = 56000 nM T52450 CP4XL8 44445237 IC50 = 39000 nM T52450 CJA79R 44445239 IC50 = 46000 nM T52450 CA72BI 44445240 IC50 = 50000 nM T52450 CZJB48 44445241 IC50 = 121000 nM T52450 C85EVH 44445242 IC50 = 135000 nM T52450 C9DI7F 44445243 IC50 = 102000 nM T52450 CVLH67 44445244 IC50 = 101000 nM T52450 CIP3X8 44445245 IC50 = 120000 nM T52450 CL1MK6 44445246 IC50 = 95000 nM T52450 C0CX7T 44445247 IC50 > 150000 nM T52450 CEZ2P7 44445248 IC50 > 150000 nM T52450 CL0K9Q 44445249 IC50 = 134000 nM T52450 C9T2SH 44445250 IC50 > 150000 nM T52450 C5EFP9 44445251 IC50 = 86000 nM T52450 CLJ71G 44445252 IC50 = 108000 nM T52450 C8TF3E 44445253 IC50 = 138000 nM T52450 C4CAY7 44445254 IC50 = 119000 nM T52450 CH1LE5 44445255 IC50 = 120000 nM T52450 CLP96W 44445256 IC50 = 92000 nM T52450 CK8S4Z 44445257 IC50 = 114000 nM T52450 C03EJW 44445258 IC50 = 124000 nM T52450 CO9SM5 44445261 IC50 = 126000 nM T52450 C3FX8B 44445262 IC50 > 150000 nM T52450 CZS8N5 44445263 IC50 > 150000 nM T52450 CMW2U6 44445264 IC50 = 99000 nM T52450 CB47AH 44445265 IC50 = 119000 nM T52450 CA43LS 44445266 IC50 = 75000 nM T52450 C23MDF 44445267 IC50 = 78000 nM T52450 C9K3DI 44445268 IC50 = 114000 nM T52450 C2ZAK4 44445269 IC50 = 108000 nM T52450 CIVC64 44445270 IC50 = 115000 nM T52450 C8W1HX 44445271 IC50 > 150000 nM T52450 CTFR27 44445272 IC50 > 150000 nM T52450 C20DNO 44445273 IC50 > 150000 nM T52450 CWLC15 44445274 IC50 > 150000 nM T52450 CZD5M3 44445275 IC50 > 150000 nM T52450 CJET46 44445276 IC50 > 150000 nM T52450 CI58AM 44445277 IC50 > 150000 nM T52450 CDN37V 44445278 IC50 > 150000 nM T52450 CE36AB 44445279 IC50 > 150000 nM T52450 CV9KX5 44445280 IC50 > 150000 nM T52450 C4S2WX 44445281 IC50 > 150000 nM T52450 C3E1PH 44445689 IC50 = 60.26 nM T52450 CSK7R8 44445690 IC50 = 338.84 nM T52450 CC6W8J 44445691 IC50 = 199.53 nM T52450 CF4N6J 44445693 IC50 = 177.83 nM T52450 CFJ1Z8 44445694 IC50 = 3467.37 nM T52450 CB61LR 44445695 IC50 = 1819.7 nM T52450 CAC3U8 44445696 IC50 = 19054.61 nM T52450 C65VFJ 44445698 IC50 = 181.97 nM T52450 CRL84B 44445699 IC50 = 338.84 nM T52450 C9TNB7 44445701 IC50 = 416.87 nM T52450 C4V7FM 44445702 IC50 = 269.15 nM T52450 CJU79N 44445703 IC50 = 851.14 nM T52450 CR78LW 44445704 IC50 = 309.03 nM T52450 CE6PV4 44445707 IC50 = 2570.4 nM T52450 C97SNB 44445708 IC50 = 2691.53 nM T52450 CMC68Z 44445709 IC50 = 1288.25 nM T52450 CN82TZ 44445710 IC50 = 218.78 nM T52450 CLBQ98 44445711 IC50 = 602.56 nM T52450 C8HD3Z 44445712 IC50 = 120.23 nM T52450 CNQ45R 44445713 IC50 = 190.55 nM T52450 CK40OY 44445714 IC50 = 1584.89 nM T52450 CEHV10 44445715 IC50 = 7762.47 nM T52450 C13HCO 44445717 IC50 = 120.23 nM T52450 C7SRW0 44445718 IC50 = 524.81 nM T52450 C8T2KM 44445720 IC50 = 1584.89 nM T52450 CPVA30 44445732 IC50 = 269.15 nM T52450 CQH24E 44445733 IC50 = 15135.61 nM T52450 CVN69U 44445734 IC50 = 10964.78 nM T52450 CY1NR2 44445735 IC50 = 5128.61 nM T52450 C80WOG 44445736 IC50 = 2187.76 nM T52450 C39OKI 44445737 IC50 = 7413.1 nM T52450 CSK38C 44445738 IC50 = 4466.84 nM T52450 C4U2VH 44445739 IC50 = 1905.46 nM T52450 CF0LB5 44445740 IC50 = 1698.24 nM T52450 CL72FG 44445741 IC50 = 2818.38 nM T52450 CH2Y7W 44445813 Ki > 10000 nM T52450 C4J2QM 44445814 Ki = 2300 nM T52450 C20HIJ 44446753 IC50 = 1892 nM T52450 C9CS8E 44446754 IC50 > 5000 nM T52450 C4Z7IQ 44446755 IC50 > 5000 nM T52450 C4K5QT 44446756 IC50 > 5000 nM T52450 C47SRV 44446758 IC50 > 5000 nM T52450 C8HM5N 44446763 IC50 > 5000 nM T52450 CU5Z4V 44446765 IC50 > 5000 nM T52450 CYO65B 44446797 IC50 > 5000 nM T52450 CH72RW 44446806 IC50 > 5000 nM T52450 CTKX08 44446807 IC50 > 5000 nM T52450 CJN1L7 44446821 IC50 > 5000 nM T52450 C4LF6Y 44446822 Ki > 4948 nM T52450 C9FG5A 44446823 IC50 > 5000 nM T52450 C1P0BV 44446824 IC50 > 5000 nM T52450 C5AW3N 44446825 IC50 > 5000 nM T52450 C17YSI 44446827 IC50 > 5000 nM T52450 CE2OM1 44446839 IC50 > 5000 nM T52450 C49VJF 44446842 IC50 > 5000 nM T52450 CF4DL2 44446843 IC50 > 5000 nM T52450 CIP23G 44447330 IC50 > 10000 nM T52450 CPS5M4 44447343 IC50 > 10000 nM T52450 CB3F0E 44447344 IC50 > 10000 nM T52450 CM7JV0 44447353 IC50 = 774 nM T52450 CY2XR5 44447363 IC50 > 10000 nM T52450 CU2BC6 44447364 IC50 > 10000 nM T52450 CD8RX4 44447437 IC50 > 5000 nM T52450 CLNK98 44447442 IC50 > 5000 nM T52450 CLNM62 44454612 IC50 > 10000 nM T52450 CZ2QY4 44454641 IC50 > 10000 nM T52450 C7DIB0 44454661 IC50 > 10000 nM T52450 CTR91D 44454664 IC50 > 10000 nM T52450 CM8AG1 44454790 IC50 > 10000 nM T52450 CCH42M 44454856 IC50 > 10000 nM T52450 CQG09B 44454861 IC50 > 10000 nM T52450 CLG57Z 44454888 IC50 > 10000 nM T52450 CMEJ96 44454891 IC50 > 10000 nM T52450 CSKN69 44455242 IC50 > 1000 nM T52450 CW46RV 44455498 Ki > 4948 nM T52450 CXNP45 44455499 Ki > 4948 nM T52450 C6CED5 44455528 Ki > 4948 nM T52450 CUQH30 44455553 Ki > 4948 nM T52450 C83KYJ 44455582 Ki > 4948 nM T52450 CK5N1S 44455612 Ki > 4948 nM T52450 CU2E7V 44455613 Ki > 4948 nM T52450 CH1DI4 44455614 Ki > 4948 nM T52450 CFQ79A 44455647 Ki > 4948 nM T52450 C3J1SV 44455676 IC50 > 1000 nM T52450 C6FV2Z 44455783 Ki > 4948 nM T52450 CPYV60 44455807 Ki > 4948 nM T52450 CGA0T4 44455829 Ki > 4948 nM T52450 C38VBL 44455836 IC50 > 1000 nM T52450 CV2B4N 44455858 Ki > 4948 nM T52450 CVR58Q 44455879 Ki > 4948 nM T52450 CWZ8K6 44455880 Ki > 4948 nM T52450 CD9N5I 44459425 Ki = 4 nM T52450 CP98IX 44459426 Ki = 2.3 nM T52450 CAM2Q6 44459443 Ki < 1 nM T52450 CVY7O1 44460358 Ki = 510 nM T52450 C78GOL 44460359 Ki = 2700 nM T52450 C4MK3N 44460370 Ki = 1000 nM T52450 CEY4L1 44460381 Ki > 10000 nM T52450 CEN93Y 44460382 Ki > 10000 nM T52450 CL30OP 44460588 Ki = 870 nM T52450 CO12NF 44460595 Ki = 1900 nM T52450 C34BMW 44460598 Ki = 3300 nM T52450 C0A1KH 44460605 Ki = 2100 nM T52450 CDN1V6 44460606 Ki = 5100 nM T52450 C8TB4H 44460611 Ki > 10000 nM T52450 CJ6PN3 44460646 Ki > 10000 nM T52450 CU8A1O 44460672 Ki > 10000 nM T52450 CIQ87B 44460676 Ki > 10000 nM T52450 C5B8NZ 44460690 Ki = 2300 nM T52450 CK4WU2 44460737 Ki > 10000 nM T52450 CY6JC5 44460927 Ki = 1500 nM T52450 CG0Z7I 44478924 IC50 > 10000 nM T52450 CFO27Y 44478926 IC50 = 4100 nM T52450 CBZJ29 44478927 IC50 = 8300 nM T52450 CRJ24K 44479197 IC50 > 10000 nM T52450 CGOH82 44479198 IC50 > 10000 nM T52450 CLV56M 44479199 IC50 = 4400 nM T52450 CY92OQ 44479458 IC50 > 200000 nM T52450 CH1QG9 44479459 IC50 = 28000 nM T52450 CB1NT7 44479460 IC50 = 29000 nM T52450 C0JQ9L 44479699 IC50 = 12000 nM T52450 C0DN1Q 44479700 IC50 > 100000 nM T52450 CTG24W 44479702 IC50 = 51000 nM T52450 CGZ49M 44479703 IC50 > 10000 nM T52450 CAK94X 44563337 IC50 = 6770 nM T52450 CSH4K3 44563364 IC50 = 330 nM T52450 CAF95R 44563365 IC50 = 5600 nM T52450 CO4FQ1 44563366 IC50 > 10000 nM T52450 C6WA3X 44563401 IC50 > 10000 nM T52450 CX5L7N 44563402 IC50 = 250 nM T52450 CJ8V4U 44563403 IC50 = 290 nM T52450 CN2BM4 44563404 IC50 = 4000 nM T52450 C3KCV6 44563405 IC50 = 5600 nM T52450 CI0R5M 44563465 IC50 = 490 nM T52450 C5IQ9Z 44563466 IC50 = 850 nM T52450 C6ZEW9 44563467 IC50 = 980 nM T52450 CZ2EL1 44563468 IC50 = 440 nM T52450 CDV6R7 44563469 IC50 = 93 nM T52450 CJ2BU5 44563487 IC50 = 150 nM T52450 C1UXP6 44563490 IC50 = 1033 nM T52450 CZ0W1A 44563491 IC50 = 2043 nM T52450 C37UAM 44563492 IC50 = 1075 nM T52450 C4BD0N 44563493 IC50 = 350 nM T52450 CNP6M7 44563494 IC50 = 110 nM T52450 CY1A8V 44564505 IC50 = 1600 nM T52450 CPT42K 44580109 IC50 > 5000 nM T52450 CQ7W5I 44580110 Ki = 5248 nM T52450 CWD32S 44580184 IC50 = 37300 nM T52450 CQ4ZR1 44580422 IC50 = 5900 nM T52450 C0XJ5C 44580496 Ki > 4949 nM T52450 CK68GT 44580539 Ki = 348 nM T52450 CXIY57 44580801 Ki > 10000000 nM T52450 C0OA8Y 44580802 Ki > 10000000 nM T52450 CNC4D7 44581071 Ki > 10000000 nM T52450 CDF48U 44581111 Ki > 10000000 nM T52450 C2Z4HB 44583600 IC50 > 5000 nM T52450 C5HA4P 44583622 IC50 > 5000 nM T52450 C7PR8I 44583623 IC50 > 5000 nM T52450 CDRC42 44583654 IC50 > 5000 nM T52450 CM79HD 44583656 IC50 > 5000 nM T52450 CS81IL 44587000 EC50 = 18.7 nM T52450 CUNV59 44587001 EC50 = 22 nM T52450 CMN58Z 44587002 EC50 = 18 nM T52450 C9RX7K 44587056 EC50 = 1.9 nM T52450 C71CKD 44587057 EC50 = 39 nM T52450 C7LU9Z 44587058 EC50 = 1.6 nM T52450 CCJ6Z0 44587059 EC50 = 83 nM T52450 C68ZVD 44587197 EC50 = 0.8 nM T52450 CF93RA 44587198 EC50 = 53.3 nM T52450 CIHA86 44587199 EC50 = 0.1 nM T52450 C68JWV 44587218 EC50 = 21 nM T52450 C2USW6 44587219 EC50 = 23.2 nM T52450 CDBQ16 44587220 EC50 = 2.8 nM T52450 CUA45E 44587248 EC50 = 1.3 nM T52450 CC0V2T 44587249 EC50 = 3.4 nM T52450 COU07A 44587250 EC50 = 21.5 nM T52450 C91YAW 44587251 EC50 = 4.9 nM T52450 CM9IN6 44592481 IC50 = 44000 nM T52450 CTW7F2 44601281 IC50 = 155 nM T52450 C0KR6J 44626353 IC50 > 98000 nM T52450 C19LWR 44634267 IC50 = 660 nM T52450 CM0I4J 45101511 IC50 > 5000 nM T52450 CACH13 45269631 IC50 = 4100 nM T52450 CH4NL1 45376336 IC50 = 3352.83 nM T52450 C3SQL2 45378250 IC50 = 1500 nM T52450 CQE49A 45378251 IC50 = 4 nM T52450 CO4AC6 45378252 IC50 = 1100 nM T52450 C42FPG 45378253 IC50 = 350 nM T52450 CI82BN 45378254 IC50 = 400 nM T52450 C6MY2W 45380188 IC50 = 1100 nM T52450 C9P0DG 45380189 IC50 = 56 nM T52450 CRY0E8 45380190 IC50 = 196 nM T52450 C0MPH3 45380191 IC50 = 5000 nM T52450 CMPE63 45482676 IC50 > 100000 nM T52450 C8AUI5 45482999 IC50 > 98000 nM T52450 C9W7IP 45483016 IC50 > 98000 nM T52450 CPB42K 45483022 IC50 > 98000 nM T52450 CBG76X 45483023 IC50 > 98000 nM T52450 CDW4C8 45483036 IC50 > 98000 nM T52450 C4ZWY7 45487310 IC50 > 5000 nM T52450 C9SV0H 45487311 IC50 > 5000 nM T52450 CCF05Q 45487333 IC50 > 5000 nM T52450 CY09ZU 45487335 IC50 > 5000 nM T52450 COX40Y 45487358 IC50 > 5000 nM T52450 CF1T7M 45487359 IC50 > 5000 nM T52450 CRXI29 45487373 IC50 > 5000 nM T52450 CYL32E 45487376 IC50 > 5000 nM T52450 CO5P9I 45487386 IC50 > 5000 nM T52450 CS9Y8G 45487387 IC50 = 2500 nM T52450 CWLC18 45487393 IC50 > 5000 nM T52450 CI4KJ5 45487400 IC50 > 5000 nM T52450 C49HOI 45487401 IC50 > 5000 nM T52450 CSX5I9 46175170 IC50 = 180 nM T52450 C56WVI 46184724 Ki > 50000 nM T52450 CZ6C8P 46703060 IC50 = 4712.73 nM T52450 C0DHL4 46703061 IC50 = 4799.42 nM T52450 CYA45K 46703062 IC50 = 4829.57 nM T52450 CY72WL 46703063 IC50 = 5247.92 nM T52450 C1YHS2 46703064 IC50 = 5285.42 nM T52450 CL2U4Z 46829322 Ki = 128 nM T52450 CH0Z1E 46844314 Ki = 176 nM T52450 C20BTY 46856241 Ki > 100000 nM T52450 C0ECU2 46861775 IC50 = 3963.66 nM T52450 C0Y9NZ 46861793 IC50 = 4366.42 nM T52450 C5L8GF 46871738 IC50 > 10000 nM T52450 CR1KF7 46871739 IC50 > 10000 nM T52450 C8Q6YR 46871740 IC50 > 10000 nM T52450 C58YSM 46871741 IC50 > 10000 nM T52450 C4VEZ3 46882679 IC50 = 4000 nM T52450 C0F7SU 46905989 IC50 = 24000 nM T52450 C49PYF 46907509 IC50 = 4246.83 nM T52450 C2U1GW 46907510 IC50 = 3706.63 nM T52450 C7MUS8 46907512 IC50 = 4302.21 nM T52450 C71YRF 46907513 IC50 = 3808.43 nM T52450 CVH58U 46907580 IC50 = 3404.64 nM T52450 C0S9WB 46919610 Ki > 100000 nM T52450 CE3H7I 46938726 IC50 = 2600 nM T52450 C9T0HR 46938727 IC50 > 10000 nM T52450 C0YR7M 46938728 IC50 > 10000 nM T52450 C2S7PK 46942365 Ki = 286 nM T52450 C7XW1Q 50907084 Ki = 32 nM T52450 C8RL5Q 50907292 Ki = 742 nM T52450 CUD7O0 50941549 IC50 > 10000 nM T52450 C7AU4S 50943150 IC50 > 100000 nM T52450 CX8N4D 50990920 IC50 > 10000 nM T52450 CXF4V3 50990921 IC50 > 19000 nM T52450 CAS94N 51346773 Ki = 41000 nM T52450 CU2SX3 51355576 Ki > 10000 nM T52450 C1Y5UN 52951473 IC50 > 10000 nM T52450 CXYJ67 52951474 IC50 > 10000 nM T52450 C8J9EM 52951589 IC50 > 10000 nM T52450 CEAS70 52951591 IC50 > 10000 nM T52450 C4DG1F 52951593 IC50 > 10000 nM T52450 C6XJ3V 52951596 IC50 > 10000 nM T52450 C9U3AF 52951710 IC50 = 3700 nM T52450 C4M1CA 52951712 IC50 > 10000 nM T52450 C76LDY 52951967 IC50 = 33 nM T52450 CYKS94 52951968 IC50 < 300 nM T52450 CE0FP3 52951969 IC50 = 1500 nM T52450 CL69OM 52951970 IC50 = 1300 nM T52450 CMPB74 52951971 IC50 = 1000 nM T52450 CZ1TN8 52951972 IC50 = 230 nM T52450 CK08OB 52952074 IC50 = 1300 nM T52450 C46AYR 52952075 IC50 > 10000 nM T52450 CR32ZW 52952076 IC50 > 10000 nM T52450 CJ9O3S 52952077 IC50 > 10000 nM T52450 C3N9TF 52952078 IC50 > 10000 nM T52450 CE4Q7F 52952273 IC50 > 10000 nM T52450 CMA69V 52952274 IC50 > 10000 nM T52450 C7KB5W 52952275 IC50 > 10000 nM T52450 CRO0X4 52952276 IC50 = 2600 nM T52450 CSJ05E 52952277 IC50 > 10000 nM T52450 C29UJB 52952388 IC50 > 10000 nM T52450 C3H5ID 52952389 IC50 > 10000 nM T52450 CSX69R 52952390 IC50 > 10000 nM T52450 CB36KP 52952492 IC50 > 10000 nM T52450 C67OEU 52952493 IC50 > 10000 nM T52450 CV1I0A 52952597 IC50 = 4200 nM T52450 CGI87K 52952598 IC50 = 2300 nM T52450 CXWI18 52952599 IC50 > 10000 nM T52450 C46VHP 52952600 IC50 > 10000 nM T52450 CH3G6R 52952601 IC50 > 10000 nM T52450 CC0Y3M 52952602 IC50 > 10000 nM T52450 CLA96C 53232689 Ki > 10000 nM T52450 C3BGW0 53233015 Ki > 40000 nM T52450 CMQZ70 53242178 IC50 > 10000 nM T52450 CB09MA 53318910 IC50 = 980 nM T52450 C47DIU 53318911 IC50 > 8100 nM T52450 CC6DR2 53318912 IC50 > 10000 nM T52450 CWH47R 53319228 Ki = 287 nM T52450 C7V1NC 53320225 IC50 > 10000 nM T52450 CVH2B7 53320226 IC50 > 70000 nM T52450 CO8QK2 53320227 IC50 > 70000 nM T52450 CTQ02K 53320639 IC50 = 4926000 nM T52450 CNS3F2 53321542 IC50 = 9700 nM T52450 C4UE6R 53322469 IC50 = 1500 nM T52450 C1N2BX 53322876 IC50 > 8000 nM T52450 CSYW40 53322877 IC50 = 55000 nM T52450 C3QHA6 53322879 IC50 > 100000 nM T52450 C1VNZ9 53324198 IC50 = 9700 nM T52450 C0H7FQ 53324260 IC50 > 10000 nM T52450 CU7YG9 53325497 IC50 > 100000 nM T52450 C4G1HK 53325498 IC50 > 10000 nM T52450 CO5L1I 53325499 IC50 > 100000 nM T52450 CZA03W 53326760 IC50 > 8500 nM T52450 CM53CG 53326761 IC50 > 79000 nM T52450 CWR6T4 53326860 IC50 > 9600 nM T52450 CPY02U 53327890 IC50 = 4800 nM T52450 CPGE80 53327891 IC50 = 2300 nM T52450 CLJ4G2 53328858 IC50 = 13000 nM T52450 C4G3QL 53328859 IC50 = 21000 nM T52450 CX1TW0 53328860 IC50 = 6700 nM T52450 C0ZX5G 53329215 IC50 = 37000 nM T52450 CSU52A 53329216 IC50 = 56000 nM T52450 CNB63X 53361475 IC50 = 108000 nM T52450 C6Y2EV 53374826 IC50 > 100000 nM T52450 CP0EC1 53375373 IC50 > 100000 nM T52450 CBL30Y 54181369 IC50 > 10000 nM T52450 CSUW40 54352406 IC50 > 5000 nM T52450 C3M8GZ 54580051 IC50 > 10000 nM T52450 CL0WM9 54580052 IC50 > 10000 nM T52450 CK26XF 54580053 IC50 > 10000 nM T52450 CS1LM9 54580054 IC50 > 10000 nM T52450 C9LD3H 54580167 Ki = 5700 nM T52450 C3LF0P 54580544 Ki > 10000 nM T52450 C6R3MZ 54580973 Ki > 50000 nM T52450 C8PE1G 54581030 IC50 > 6700 nM T52450 CZD7Y6 54581162 Ki = 32000 nM T52450 CVO09J 54581546 Ki = 3700 nM T52450 CWKA42 54582019 Ki = 33000 nM T52450 CVK72M 54582073 IC50 > 10000 nM T52450 CBK18O 54582074 IC50 > 10000 nM T52450 CP2F1B 54582075 IC50 > 10000 nM T52450 CZNU23 54582076 IC50 > 10000 nM T52450 C0U5HZ 54582077 IC50 > 10000 nM T52450 CSTG96 54582078 IC50 > 10000 nM T52450 C8SG9Y 54582079 IC50 > 10000 nM T52450 CZI6S3 54582080 IC50 > 10000 nM T52450 CW6VD0 54582183 Ki = 6700 nM T52450 CD09BZ 54582543 Ki > 10000 nM T52450 CH6Q2Z 54583016 IC50 > 10000 nM T52450 C3V9LQ 54583017 IC50 > 10000 nM T52450 CT80KQ 54583018 IC50 > 10000 nM T52450 CPT4L5 54583019 IC50 > 10000 nM T52450 C8N4YL 54583153 Ki = 27000 nM T52450 CK52YD 54583511 Ki > 10000 nM T52450 CBEV27 54584024 IC50 > 10000 nM T52450 CM87DP 54584025 IC50 > 10000 nM T52450 CIT0S7 54584142 Ki = 16000 nM T52450 C86WVF 54584143 Ki = 50000 nM T52450 C8UL3W 54585079 Ki = 25000 nM T52450 C28GKQ 54585927 IC50 > 10000 nM T52450 C3P4KW 54586055 Ki = 120000 nM T52450 CAZ76E 54586892 IC50 > 10000 nM T52450 CM0OQ3 54586893 IC50 > 10000 nM T52450 CK1NS7 54586894 IC50 > 10000 nM T52450 CMC4Y1 54586895 IC50 > 10000 nM T52450 C2MKX5 54586896 IC50 > 10000 nM T52450 CU91QP 54586897 IC50 > 10000 nM T52450 CI08RQ 54586898 IC50 > 10000 nM T52450 C6PRI4 54586899 IC50 > 10000 nM T52450 CG37UX 54587429 Ki > 10000 nM T52450 CL9SC3 54587769 Ki > 40000 nM T52450 CGH0S7 54589400 IC50 > 100000 nM T52450 C83NUI 54687474 IC50 > 50000 nM T52450 CZ6V0U 54724681 IC50 > 50000 nM T52450 CJ6HT4 54726662 IC50 = 30000 nM T52450 C9P5ES 54752445 IC50 > 1000 nM T52450 C0HKC9 54752446 IC50 > 1000 nM T52450 C6D9IE 54753443 IC50 = 3570.27 nM T52450 C5D1TI 56649332 IC50 > 1000 nM T52450 CKJ9S1 56835167 IC50 = 1600 nM T52450 C21CLZ 56835168 IC50 = 1300 nM T52450 C0L2TS 56835169 IC50 = 4900 nM T52450 C7FQY9 57125118 IC50 = 227 nM T52450 C10BMZ 57127110 IC50 > 10000 nM T52450 CQU16V 57339411 Ki = 5700 nM T52450 C6LM3B 57339412 Ki = 1800 nM T52450 CHE2I1 57345500 Ki > 50000 nM T52450 C63TFM 57345501 Ki > 50000 nM T52450 C8KT2F 57345502 Ki = 47000 nM T52450 C0KPD8 57384084 IC50 = 4000 nM T52450 CV67JB 57384091 IC50 = 2500 nM T52450 CR8MW2 57391205 IC50 > 10000 nM T52450 CP5BX6 57394607 IC50 > 1000 nM T52450 CNOH63 57394711 IC50 > 10000 nM T52450 CE5X3D 57394850 IC50 > 50000 nM T52450 CG43ME 57394903 IC50 = 1000 nM T52450 CWH7V8 57561293 IC50 = 4710 nM T52450 CY1N3J 57792153 IC50 = 1132 nM T52450 CCKD80 58307579 Ki = 850 nM T52450 CX73PT 59033102 IC50 > 25000 nM T52450 CAT67H 59910477 IC50 > 10000 nM T52450 CLZ72F 70682077 IC50 = 340 nM T52450 C8B6WD 70688393 IC50 = 8230 nM T52450 C6P3XM 70693710 Ki > 50000 nM T52450 C0HE2P 70694634 IC50 = 3250 nM T52450 CL7JF9 71304794 IC50 = 11800 nM T52450 CSY30R 71304795 IC50 = 280 nM T52450 CNPG78 71304796 IC50 = 16000 nM T52450 CI8X5B 71449151 IC50 = 2530 nM T52450 CMW3O0 71451330 Ki > 200 nM T52450 C9QS6E 71456659 Ki > 2000 nM T52450 C2OL0I 71457963 IC50 = 1800 nM T52450 CYB60V 71458014 IC50 = 800 nM T52450 C9RE0A 71559535 IC50 = 3602.31 nM T52450 C47TMN 71559652 IC50 = 3595.63 nM T52450 CN2XB4 71559653 IC50 = 5207.75 nM T52450 CZHQ79 71559654 IC50 = 5275.93 nM T52450 CO59LK 71559762 IC50 = 5206.82 nM T52450 CGL35Z 71559763 IC50 = 5127.23 nM T52450 C7U5LE 71559764 IC50 = 5162.55 nM T52450 CD6L1J 71559765 IC50 = 5219.32 nM T52450 CXKO04 71559766 IC50 = 4741.38 nM T52450 CA14SK 71559767 IC50 = 4767.79 nM T52450 COZ56A 71559768 IC50 = 4117.53 nM T52450 CZ9X1J 71559769 IC50 = 4213.83 nM T52450 C5NHI1 71559770 IC50 = 4387.42 nM T52450 CF9JE8 71559897 IC50 = 3496.65 nM T52450 CGT96R 71559898 IC50 = 5058.56 nM T52450 C01PTX 71559899 IC50 = 5347.73 nM T52450 C96OCB 71559900 IC50 = 5114.38 nM T52450 CJB0D9 71559901 IC50 = 5217.29 nM T52450 C6Y1IE 71559902 IC50 = 5293.55 nM T52450 C24ZYC 71559903 IC50 = 4788.43 nM T52450 CC3MY7 71559904 IC50 = 4879.72 nM T52450 C7WMU5 71560026 IC50 = 4233.53 nM T52450 C60VEX 71560027 IC50 = 4426.63 nM T52450 CN1VF7 71560028 IC50 = 4538.24 nM T52450 CSY3D5 71560029 IC50 = 3574.82 nM T52450 CH5J4A 71602247 IC50 = 18500 nM T52450 CH53IU 71602248 IC50 = 11500 nM T52450 C97EWQ 71602249 IC50 = 6100 nM T52450 CVDB83 71652189 IC50 = 38900 nM T52450 CCTS74 71652190 IC50 = 41700 nM T52450 C5SVH1 71652191 IC50 = 42600 nM T52450 CWYV26 71652192 IC50 = 10700 nM T52450 C84OUA 71652193 IC50 = 34700 nM T52450 CSA5O8 71652194 IC50 = 38500 nM T52450 CL3NU8 71652195 IC50 = 8600 nM T52450 CNX9B1 71652215 IC50 > 5000 nM T52450 C7RZN9 71652216 IC50 = 27000 nM T52450 CL6V4Y 71652358 IC50 = 8900 nM T52450 CUXZ29 71652359 IC50 > 100000 nM T52450 CE5W0J 71652360 IC50 = 13700 nM T52450 CS3A5U 71652361 IC50 = 2500 nM T52450 CX1F0N 71652362 IC50 > 100000 nM T52450 CK93HG 71652363 IC50 > 100000 nM T52450 C0NTU7 71652382 IC50 = 2900 nM T52450 CA5XS1 71652383 IC50 > 5000 nM T52450 C6ET4B 71652522 IC50 = 7600 nM T52450 CPKF31 71652523 IC50 = 5500 nM T52450 C6DA0U 71652524 IC50 = 3600 nM T52450 CB95AO 71652525 IC50 = 4200 nM T52450 C6VU1O 71652526 IC50 = 6800 nM T52450 CA97QZ 71652527 IC50 = 10600 nM T52450 CYS46I 71652677 IC50 = 400 nM T52450 CN5A7P 71654192 IC50 > 100000 nM T52450 CYQM29 71654194 IC50 > 100000 nM T52450 CUDA81 71654195 IC50 > 100000 nM T52450 C5KYI7 71654355 IC50 > 100000 nM T52450 CH81YW 71654357 IC50 > 100000 nM T52450 CX67VE 71654516 IC50 = 800 nM T52450 CU01TG 71654517 IC50 = 53700 nM T52450 CKO45B 71654518 IC50 > 100000 nM T52450 C6KEH0 71680708 Ki = 25000 nM T52450 C7DMX5 71680709 Ki = 4100 nM T52450 CFPM82 71680710 Ki = 2800 nM T52450 C9ZOM7 71680866 Ki > 3000 nM T52450 CQ68LT 71680868 Ki > 50000 nM T52450 CFH2V0 71681183 Ki = 6300 nM T52450 CV3X1T 71682766 Ki > 100000 nM T52450 C80EYX 71682913 Ki > 20000 nM T52450 CIBD03 71682914 Ki = 10000 nM T52450 C41BYG 71682915 Ki = 2100 nM T52450 CQ29PJ 71682917 Ki > 200000 nM T52450 CFWN65 71683062 Ki > 200000 nM T52450 CM4E5A 71716445 IC50 = 4831.49 nM T52450 C45PSZ 71717046 IC50 = 3448.67 nM T52450 C9Z4PI 71718276 IC50 = 3401.82 nM T52450 C2XW5I 71718291 IC50 = 3256.49 nM T52450 C18RDB 71719502 IC50 = 4889.64 nM T52450 CR28AW 71734195 IC50 > 1000 nM T52450 C50SID 71817098 Ki = 19700 nM T52450 C7YFC8 72711513 IC50 > 500000 nM T52450 CTM4P2 72713638 IC50 = 120000 nM T52450 C0N2JX 72713639 IC50 = 32000 nM T52450 CF4K8Y 72713862 IC50 = 74000 nM T52450 C3R6JO 72713863 IC50 > 500000 nM T52450 CW9D3V 72713864 IC50 > 500000 nM T52450 CQ6FH3 72713865 IC50 = 61000 nM T52450 C4FYB0 72713866 IC50 > 500000 nM T52450 CH6SI1 72713867 IC50 = 100000 nM T52450 CS21QM 72713868 IC50 = 620000 nM T52450 CB56AP 72714081 IC50 = 181000 nM T52450 C1CK0E 72714082 IC50 > 500000 nM T52450 CP5Q8W 72714083 IC50 > 200000 nM T52450 CRUH64 72714085 IC50 > 200000 nM T52450 CZFY06 72714322 IC50 = 400000 nM T52450 CDY70J 72714323 IC50 = 370000 nM T52450 CD56BA 72714324 IC50 > 500000 nM T52450 CTOQ24 73054451 IC50 > 100000 nM T52450 CK9TU0 73055013 IC50 > 100000 nM T52450 C7UQ1B 73055016 IC50 > 100000 nM T52450 CO5FN4 73055018 IC50 > 100000 nM T52450 C8H0UN 73055605 IC50 > 100000 nM T52450 C01SHT 73055902 IC50 = 78000 nM T52450 C2GE8Q 73055903 IC50 > 100000 nM T52450 CDA75O 73055905 IC50 > 100000 nM T52450 CK5FT8 73055906 IC50 > 100000 nM T52450 C9OX6Y 73055907 IC50 > 100000 nM T52450 CA93JD 73056179 IC50 = 50000 nM T52450 CEX86T 73056180 IC50 = 65000 nM T52450 C8QZG6 73056181 IC50 > 100000 nM T52450 C1KGT9 73056183 IC50 > 100000 nM T52450 CR75BY 73056185 IC50 > 100000 nM T52450 C7YT0C 73056773 IC50 > 100000 nM T52450 C46YCT 73345375 Ki = 13000 nM T52450 C38IDL 73345835 Ki = 52 nM T52450 CE05UK 73347034 Ki = 3180 nM T52450 CTP71B 73348406 Ki = 22000 nM T52450 CR3HX8 73348408 Ki = 240000 nM T52450 C9W7OB 73348532 Ki = 2900 nM T52450 CW01EA 73349535 IC50 > 10000 nM T52450 CX86VY 73349984 Ki = 130000 nM T52450 C8ROG3 73350414 Ki = 99 nM T52450 CF7AB2 73350415 Ki = 110 nM T52450 C54FRN 73351483 Ki = 29000 nM T52450 C2PFM4 73351930 Ki = 260 nM T52450 CVP75M 73352951 Ki = 49000 nM T52450 CI18HF 73353270 Ki = 19000 nM T52450 CC7OE8 73354605 Ki = 820 nM T52450 CX6S3Y 73354606 Ki = 370 nM T52450 CGS1Q4 73354607 IC50 = 5900 nM T52450 C4X9OZ 73354608 Ki = 1740 nM T52450 CI09CY 73354906 Ki = 75 nM T52450 C6H5TU 73354941 Ki = 7000 nM T52450 CUB7V9 76329513 IC50 = 150 nM T52450 C21FEO 76331549 IC50 = 522 nM T52450 CX39OW 76331563 IC50 = 6480 nM T52450 C9CY5K 76335167 IC50 = 1140 nM T52450 CGQ8F3 86287515 IC50 = 11000 nM T52450 CJ37XE 86287516 IC50 = 19000 nM T52450 COV8I9 86291010 IC50 = 1059 nM T52450 C8FGM5 90663041 IC50 = 460 nM T52450 CG3E4Y 90663043 IC50 = 307 nM T52450 CYX8F2 90663045 IC50 = 2230 nM T52450 CH8V6R 90663046 IC50 = 510 nM T52450 CVPH63 90663059 Ki = 22000 nM T52450 C6AK3O 90663060 Ki = 29000 nM T52450 CUZD67 90663061 Ki = 14000 nM T52450 CTQ17J 90663062 Ki = 72000 nM T52450 CQGJ90 90663063 Ki = 9000 nM T52450 C0ZH1K 90663064 Ki = 19000 nM T52450 CD53CF 90663065 Ki = 19000 nM T52450 C1A4QT 90663067 Ki = 19000 nM T52450 CLW7Q8 90663069 Ki = 33000 nM T52450 C6JY4Q 90663070 Ki = 80000 nM T52450 C7YU1I 90663071 Ki = 19000 nM T52450 C07RTW 90663072 Ki = 13000 nM T52450 CZ68QM 90663073 Ki = 28000 nM T52450 CVTJ63 90663074 Ki = 15000 nM T52450 C9J8HB 90663075 Ki = 10000 nM T52450 C06GRV 90663076 Ki = 12000 nM T52450 CF2L9A 90663077 Ki = 87000 nM T52450 CGL0N7 90663078 Ki = 18000 nM T52450 COP05M 90663079 Ki = 14000 nM T52450 C1E5CB 90663080 Ki = 69000 nM T52450 C6IXP4 90663081 Ki = 74000 nM T52450 C0S7NT 90663082 Ki = 15000 nM T52450 C8MOY6 90663083 Ki = 30000 nM T52450 C4NP9W 90663084 Ki = 24000 nM T52450 CD3C8E 90663085 Ki = 20000 nM T52450 C63NOF 90663086 Ki = 24000 nM T52450 CU3LC2 90663087 Ki = 21000 nM T52450 CQ9C5I 90667651 IC50 > 50000 nM T52450 CGXO89 90667652 IC50 > 50000 nM T52450 CMG37C 91867803 Ki = 270000 nM T52450 CRT54C 101910871 IC50 = 100000 nM T52450 C1J3CK 117094707 IC50 = 346000 nM T52450 C1W5NH 118718816 IC50 = 3200 nM T52450 CHXB96 118723754 IC50 = 40 nM T52450 CJFS09 122190237 IC50 = 26000 nM T52450 C9QKI3 127020966 IC50 > 100000 nM T52450 CT03QA 127026888 IC50 > 200000 nM T52450 C89QOM 127043503 IC50 > 10000 nM T52450 C9E5YJ 127043505 IC50 > 10000 nM T52450 CW1Q3D 127043506 IC50 > 10000 nM T52450 C1C7WB 127044036 IC50 > 10000 nM T52450 CPF6U7 127044139 IC50 > 10000 nM T52450 CT9B0Q 127044462 IC50 > 10000 nM T52450 CL3X1A 127044649 IC50 > 10000 nM T52450 C8RZ7T 127044651 IC50 > 10000 nM T52450 C3I4PT 127044652 IC50 > 10000 nM T52450 CDX86T 127044818 IC50 > 10000 nM T52450 C56OJV 127044819 IC50 > 10000 nM T52450 CYA92R 130282633 IC50 = 4500 nM T52450 CO3QE2 130282636 IC50 = 4600 nM T52450 CTN42D 132941363 IC50 = 100000 nM T52450 C83FAY 134130294 Ki = 143 nM T52450 CT3G2U 134133460 IC50 = 13 nM T52450 C8VLY0 134144890 IC50 = 2050 nM T52450 C93ZLI 134145328 IC50 = 1600 nM T52450 C7K4PA 135412054 IC50 > 40000 nM T52450 C31VAN 135412231 IC50 > 40000 nM T52450 CHV2U1 135438561 IC50 > 10000 nM T52450 CRAZ20 135485671 IC50 = 1.3 nM T52450 C2URS4 135501193 IC50 = 330 nM T52450 C8R4FB 135546884 IC50 > 40000 nM T52450 C1MOD4 135567320 IC50 > 5000 nM T52450 CA5JR6 136054481 IC50 > 10000 nM T52450 CV47JN 136054485 IC50 > 10000 nM T52450 CZ48WO 136054487 IC50 > 10000 nM T52450 C8FGT0 136054495 IC50 > 10000 nM T52450 CG70BZ 136054516 IC50 = 18 nM T52450 CSM57W 136054520 IC50 > 10000 nM T52450 CTY79S 136118013 Ki > 4946 nM T52450 CTE87J 136118014 Ki > 4946 nM T52450 CIEW62 136380958 IC50 = 3400 nM T52450 C9HS7J 137287436 IC50 = 11 nM T52450 C0I6RH 137632487 IC50 = 64 nM T52450 C4UMY5 137636781 IC50 > 5000 nM T52450 CR8H9Z 137644167 IC50 > 5000 nM T52450 CB8M6U 137646865 IC50 > 5000 nM T52450 CK4LE6 137647628 IC50 > 10000 nM T52450 CZB75K 137657128 IC50 > 10000 nM T52450 CC3I9B 137660260 IC50 = 4000 nM T52450 CAB7Q6 137660566 IC50 > 10000 nM T52450 C4H0EM 137661370 IC50 > 5000 nM T52450 CZ8H6N 137661550 IC50 = 50000 nM T52450 C1Q2BP 145949247 IC50 > 5000 nM T52450 C6TD4M 145949288 IC50 > 5000 nM T52450 CN9RD6 145949408 IC50 > 5000 nM T52450 C5FWA2 145949488 IC50 > 5000 nM T52450 CZS1N7 145949693 IC50 > 5000 nM T52450 C6IPV3 145949783 IC50 > 500000 nM T52450 CYG32L 145950058 IC50 > 5000 nM T52450 C72LGN 145950074 IC50 > 500000 nM T52450 CU53BP 145950331 IC50 > 5000 nM T52450 CY8C4A 145950332 IC50 > 5000 nM T52450 CAJ25P 145951291 IC50 > 5000 nM T52450 C3EF7N 145952515 IC50 > 5000 nM T52450 CW1GS2 145952760 IC50 > 5000 nM T52450 CFN1R7 145952843 IC50 > 5000 nM T52450 CM6T2O 145953417 IC50 > 5000 nM T52450 C6FYK8 145953609 IC50 > 5000 nM T52450 CV80WQ 145954107 IC50 > 5000 nM T52450 C16VNH 145954604 IC50 > 5000 nM T52450 CQF50V 145954863 IC50 > 5000 nM T52450 C2HAG8 145955226 IC50 > 500000 nM T52450 C8QW9G 145955776 IC50 > 5000 nM T52450 CH0ZO5 145955778 IC50 > 5000 nM T52450 CFDZ62 145955866 IC50 > 5000 nM T52450 CVZ5U7 145955868 IC50 > 5000 nM T52450 C8TPR1 145956198 IC50 > 5000 nM T52450 COR96H 145956298 IC50 > 500000 nM T52450 CR8U7Y 145956318 IC50 > 5000 nM T52450 C7R3FE 145956426 IC50 > 500000 nM T52450 C4S8LU 145956764 IC50 > 5000 nM T52450 CUS0Y9 145957234 IC50 > 5000 nM T52450 CUO69Q 145957392 IC50 > 5000 nM T52450 CX94UK 145957493 IC50 > 5000 nM T52450 C6MHN7 145957508 IC50 > 5000 nM T52450 CQ15DP 145957734 IC50 > 500000 nM T52450 C5K7PV 145958060 IC50 > 5000 nM T52450 CBE02W 145958354 IC50 > 5000 nM T52450 CQL4O0 145959327 IC50 > 5000 nM T52450 CG03OE 145959777 IC50 > 500000 nM T52450 CIQ9J2 145960035 IC50 > 500000 nM T52450 CUAT97 145960347 IC50 > 5000 nM T52450 CZ76WA 145962290 IC50 > 5000 nM T52450 C27MTZ 145962695 IC50 > 5000 nM T52450 CRY63E 145963538 IC50 > 5000 nM T52450 CVCL61 145963739 IC50 > 5000 nM T52450 CWY5X0 145971805 IC50 > 10000 nM T52450 C1FPG2 145972660 IC50 > 5000 nM T52450 CJF73O 145973630 IC50 > 5000 nM T52450 CX7M9L 145976456 IC50 > 5000 nM T52450 C1KPL5 145976497 IC50 = 260000 nM T52450 CPD1B0 145977213 IC50 > 5000 nM T52450 C9Z5DX 145978402 IC50 > 5000 nM T52450 CZ25LW 155512044 IC50 = 100000 nM T52450 C98HMU 155515777 IC50 = 870 nM T52450 CRY3D4 155541376 IC50 = 150 nM T52450 CH40UO 155562232 IC50 = 45 nM T52450 CU42CE 155567829 IC50 > 100000 nM T52450 CLT4Y6 10138589 Ki = 260 nM T52450 CV4TJ8 11794277 Ki = 15000 nM T52450 D00KSS 18411961 IC50 > 10000 nM T52450 D01OCR 19366856 IC50 = 600 nM T52450 D01QOB 44404479 IC50 = 920 nM T52450 D02BTV 9816867 IC50 = 93 nM T52450 D02EFQ 10549609 IC50 = 6200 nM T52450 D02PKO 44294636 IC50 > 10000 nM T52450 D02UYR 9907830 Ki = 2 nM T52450 D03AMR 9849669 Ki = 21 nM T52450 D03FEI 15516781 IC50 > 10000 nM T52450 D03QAN 71166 IC50 = 31000 nM T52450 D03WJG 9910222 Ki = 8 nM T52450 D04GOO 10111838 IC50 > 100000 nM T52450 D04UBY 45483018 IC50 > 98000 nM T52450 D04VPH 45376872 IC50 > 22000 nM T52450 D04WWO 9889867 Ki > 4949 nM T52450 D05PTT 5281792 IC50 = 5600 nM T52450 D05THD 44478925 IC50 = 73000 nM T52450 D06BYR 44404478 IC50 = 22 nM T52450 D06EHW 11625778 IC50 > 5000 nM T52450 D07DRT 46175162 Ki > 6000 nM T52450 D07GEL 10344307 Ki = 3 nM T52450 D07MJD 44479701 IC50 = 23000 nM T52450 D08ELY 9838786 IC50 = 110 nM T52450 D08ZDD 44404461 Ki = 33 nM T52450 D09GIL 66160 IC50 > 2000 nM T52450 D09GLA 4368 IC50 = 143 nM T52450 D09SYW 44404537 IC50 = 22 nM T52450 D09XUQ 19366844 IC50 = 1500 nM T52450 D09ZOA 25049753 Ki = 365 nM T52450 D0A0FY 44479457 IC50 > 100000 nM T52450 D0A4TC 446504 IC50 = 2.5 nM T52450 D0B3UN 44580458 Ki = 67000 nM T52450 D0BI8T 44288042 IC50 = 6.9 nM T52450 D0C1EQ 20348772 IC50 > 98000 nM T52450 D0D7UA 10267279 IC50 = 1500 nM T52450 D0F4UT 21496278 IC50 > 98000 nM T52450 D0F7BE 4369084 Ki = 31000 nM T52450 D0G3YZ 11391583 IC50 > 98000 nM T52450 D0H2PA 9886977 Ki = 1 nM T52450 D0H6CK 10160968 Ki > 4949 nM T52450 D0K0YX 44626352 IC50 > 98000 nM T52450 D0K3RC 44294677 IC50 = 1700 nM T52450 D0K4TI 49292 IC50 > 2000 nM T52450 D0L6ND 10089677 IC50 = 2 ug.mL-1 T52450 D0LB0N 45483008 IC50 > 98000 nM T52450 D0LL8I 9830392 IC50 > 10000 nM T52450 D0LM2K 45483015 IC50 > 98000 nM T52450 D0N0FX 19366816 IC50 = 1000 nM T52450 D0N6CD 10565532 IC50 = 54 nM T52450 D0N8YA 159596 IC50 = 2000 nM T52450 D0NP8A 10370504 IC50 = 51000 nM T52450 D0NV9C 22004198 IC50 = 270 nM T52450 D0P2OA 47697 Ki = 33 nM T52450 D0P2TS 9818682 IC50 > 10000 nM T52450 D0Q4TA 10044321 IC50 = 2900 nM T52450 D0Q9LC 44385624 IC50 > 2000 nM T52450 D0R2BO 194777 IC50 = 3 nM T52450 D0S9OL 10155934 IC50 > 10000 nM T52450 D0T1FR 44457233 IC50 > 100000 nM T52450 D0T4AN 44404521 IC50 = 920 nM T52450 D0TL3N 45482998 IC50 > 98000 nM T52450 D0V9EN 689043 IC50 = 238.91 nM T52450 D0VI2A 44447430 IC50 = 4999 nM T52450 D0W2UK 6914621 Ki = 30000 nM T52450 D0W3ME 4369080 Ki = 3000 nM T52450 D0XE4B 15516780 IC50 = 8000 nM T52450 D0XK7G 10445302 Ki = 33 nM T52450 D0Y5IQ 44255320 IC50 = 5000 nM T52450 D0Y7NV 2220392 IC50 > 2000 nM T52450 D0YN1A 893637 Ki = 29000 nM T52450 D0Z7EF 2777 IC50 > 10000 nM T00645 D03HUX 49792852 IC50 > 10000 nM T00645 D07HPJ 11476171 IC50 > 10000 nM T00645 D09IYM 24905401 IC50 < 10 nM T00645 D09XZL 56962369 IC50 < 1 nM T00645 D0E3TC 44259 IC50 = 1.58 nM T00645 D0O0LS 25141092 IC50 > 10000 nM T00645 D0P1CV 46191454 IC50 > 10000 nM T00645 D0Q9UX 16718576 IC50 > 10000 nM T00645 D0R2TM 5287736 IC50 = 50 nM T00645 C3FD6V 13028 IC50 > 100000 nM T00645 CP9AM1 599038 Ki = 960 nM T00645 CE2G1Z 607858 Ki = 380 nM T00645 CN8SU3 684961 Ki > 3300 nM T00645 C5LHO7 753058 Ki > 4000 nM T00645 CSE25J 2123970 Ki > 5000 nM T00645 C5O3TE 4801910 Ki > 5000 nM T00645 CI4DE0 4803142 Ki = 1400 nM T00645 C6AD8F 5038004 Ki = 1100 nM T00645 CLA43B 5327919 IC50 = 1400 nM T00645 CPDC54 5327920 IC50 = 350 nM T00645 CCB9G3 5327921 IC50 = 70 nM T00645 CRTQ98 5327922 IC50 = 30 nM T00645 CWN6P7 5702541 IC50 = 100 nM T00645 CHQ7M1 8123789 Ki = 2000 nM T00645 CQV9N0 8123825 Ki = 2090 nM T00645 C2UGV9 10030483 IC50 = 450 nM T00645 CG7JO8 10099482 IC50 = 7500 nM T00645 C93LPQ 10099652 IC50 = 1700 nM T00645 CF9A5O 10125353 Ki = 1400 nM T00645 CM79VS 10149184 Ki > 3300 nM T00645 CC8XJ5 10171595 Ki = 1300 nM T00645 CB28QI 10171783 Ki > 5000 nM T00645 CJ39UQ 10236371 Ki = 600 nM T00645 CEH41V 10392789 IC50 = 170 nM T00645 C87AML 10402473 Ki > 5000 nM T00645 C7HBP6 10429593 IC50 > 10000 nM T00645 C10PAC 10460251 IC50 = 230 nM T00645 CX7S8N 10482293 IC50 = 50 nM T00645 C76QGP 10506540 IC50 = 250 nM T00645 CDNP37 10530708 IC50 = 220 nM T00645 C5EYJ3 10554684 IC50 = 5200 nM T00645 C71UIS 10555532 IC50 = 38000 nM T00645 C5YMK8 10769011 IC50 = 90 nM T00645 C5R7EZ 10901296 IC50 = 430 nM T00645 CS2YO1 11492918 Ki = 1200 nM T00645 C71WAD 11615485 Ki > 3300 nM T00645 C65FVB 11694317 Ki > 3300 nM T00645 C9JT4S 11847343 IC50 = 332 nM T00645 CHR92S 11858109 IC50 > 100000 nM T00645 CW53JC 11998038 Ki = 110 nM T00645 C90OYV 14044888 IC50 > 100000 nM T00645 CC9RM5 16344190 Ki = 3500 nM T00645 C5XFD3 17757326 Ki > 3300 nM T00645 CV78RB 18581471 Ki = 1580 nM T00645 CL81VC 21100709 IC50 = 100000 nM T00645 CLG9Z8 23366090 IC50 > 50000 nM T00645 CKYB29 23644745 IC50 = 32000 nM T00645 CMK3N9 24180453 IC50 = 168000 nM T00645 C7YG1N 24759534 IC50 = 15000 nM T00645 CQNP54 24764449 IC50 = 100000 nM T00645 C4Z9CN 24769780 IC50 > 25000 nM T00645 CZI9P0 24829572 Ki > 3300 nM T00645 C4T3UC 24829746 Ki > 3300 nM T00645 C47LFZ 24830567 Ki = 780 nM T00645 C9E7AU 24830568 Ki = 2200 nM T00645 CJ4K3P 24830569 Ki > 3300 nM T00645 CKL92Z 24830570 Ki = 140 nM T00645 C2K1OE 24830571 Ki = 3000 nM T00645 CP4KZ1 24830882 Ki = 850 nM T00645 C4J6AD 24831672 Ki > 3300 nM T00645 C82YBD 24831841 Ki > 3300 nM T00645 CTXJ06 24832008 Ki > 3300 nM T00645 C75KOR 24832012 Ki = 1850 nM T00645 C4EG8R 24993189 IC50 > 10000 nM T00645 C5WQD6 25141061 IC50 = 2600 nM T00645 C2DFB6 25189112 IC50 > 100000 nM T00645 CSY93F 25190765 IC50 = 26000 nM T00645 C0BCX6 25190766 IC50 = 2100 nM T00645 C19TVC 25190767 IC50 = 54 nM T00645 CK9V3Y 25190768 IC50 = 13.4 nM T00645 CD7S6Q 25190770 IC50 = 97 nM T00645 C3HU6A 25190771 IC50 = 21.1 nM T00645 C0CXM8 25190790 IC50 = 8.3 nM T00645 CNG96H 25210579 IC50 > 10000 nM T00645 C0K2NM 41107723 Ki > 5000 nM T00645 C75GFD 42633960 Ki = 30 nM T00645 C13TNU 44315122 IC50 = 2600 nM T00645 C3YN1R 44315123 IC50 = 3600 nM T00645 CPJ57U 44315124 IC50 < 330 nM T00645 C9HA8T 44315171 IC50 = 130 nM T00645 C2T3VN 44315184 IC50 = 26000 nM T00645 C3SP0H 44315423 IC50 = 3000 nM T00645 C8OAE9 44315457 IC50 = 4500 nM T00645 C3JS6X 44315503 IC50 = 1900 nM T00645 CEZ68T 44315545 IC50 = 13000 nM T00645 CF8B2Z 44417818 IC50 = 5.3 nM T00645 CNAB39 44435670 IC50 > 1000000 nM T00645 CNQ1E4 44435671 IC50 = 97.3 nM T00645 CJP46E 44435672 IC50 = 12.88 nM T00645 CDN3C4 44622839 Ki = 2800 nM T00645 C5G0UA 44622840 Ki = 34 nM T00645 CAZE46 46175126 IC50 = 14 nM T00645 C3HG7B 46882134 IC50 = 390 nM T00645 CTSE94 46882135 IC50 = 61 nM T00645 CSY9H1 46882136 IC50 = 3250 nM T00645 CO16JL 46882137 IC50 = 5.5 nM T00645 CJEM76 46882138 IC50 = 4.9 nM T00645 CRZ91X 46882835 IC50 = 183000 nM T00645 CS0V9G 46882836 IC50 = 23000 nM T00645 CU8WX3 46882837 IC50 = 240000 nM T00645 CNTS27 46883044 Ki = 540 nM T00645 C0DB5Z 46883045 Ki = 720 nM T00645 C9WE4S 46883122 Ki > 5000 nM T00645 CNTS75 46883123 Ki > 5000 nM T00645 CJS68B 46883124 Ki > 5000 nM T00645 CU3O2G 46883125 Ki > 4000 nM T00645 CH9RV4 46883165 Ki = 2500 nM T00645 CT1K6A 46883166 Ki > 3300 nM T00645 CGZ1S4 46883167 Ki > 3300 nM T00645 C2VGJ9 46883168 Ki = 2600 nM T00645 CT5V8K 46883169 Ki = 1500 nM T00645 CHSF07 49806372 IC50 > 1000 nM T00645 CF91RS 49843531 IC50 > 10000 nM T00645 C2Y6QS 50938552 IC50 > 10000 nM T00645 C9NYP4 51036677 IC50 > 10000 nM T00645 C4WRY3 51037112 IC50 > 10000 nM T00645 CRI28Z 51037948 IC50 > 10000 nM T00645 C2W9OA 53324451 IC50 > 10000 nM T00645 C0SWH5 53348216 IC50 > 40000 nM T00645 CE1ZK6 54759168 IC50 > 10000 nM T00645 CM8JX1 56604907 IC50 = 100000 nM T00645 CXJ63M 59603829 IC50 > 100000 nM T00645 CQEU96 59603842 IC50 = 27 nM T00645 CE37AG 60097359 Ki = 2900 nM T00645 CGUC54 60097393 Ki > 4000 nM T00645 C5MDR3 60097396 Ki = 1070 nM T00645 CGI82D 60097406 Ki = 1700 nM T00645 COH62U 60097413 Ki > 4000 nM T00645 CFMP63 60097457 Ki > 4000 nM T00645 CPO71M 60097461 Ki > 4000 nM T00645 CVD9Y1 60097467 Ki > 4000 nM T00645 CJ5V4X 60097469 Ki > 4000 nM T00645 CYC65S 60097478 Ki = 1700 nM T00645 C1MR8Q 60097495 Ki > 4000 nM T00645 CZT2A8 60097525 Ki = 580 nM T00645 C7DP4E 60097576 Ki > 5000 nM T00645 CMF42W 60097605 Ki = 600 nM T00645 C31NRA 60097624 Ki > 4000 nM T00645 CP5B0G 60097630 Ki > 3300 nM T00645 C8LYG4 60097631 Ki > 4000 nM T00645 CW1AE2 60097642 Ki = 2300 nM T00645 CO27YK 60097661 Ki > 5000 nM T00645 C2C3DJ 60097665 Ki = 2400 nM T00645 C02BUA 60097693 Ki > 5000 nM T00645 C96PLJ 60097708 Ki > 5000 nM T00645 C2VG1E 60097724 Ki > 5000 nM T00645 CS73TH 60097732 Ki = 520 nM T00645 CK6WO0 66552478 IC50 < 10000 nM T00645 C1HSE0 67035086 IC50 = 780 nM T00645 CWI6K5 67035106 IC50 > 10000 nM T00645 C38RGB 67035556 IC50 > 10000 nM T00645 C8I7GC 68293638 IC50 > 10000 nM T00645 CD56XK 68293660 IC50 > 10000 nM T00645 C5DGR9 69036886 IC50 = 10000 nM T00645 CHM7O3 72946668 IC50 > 100000 nM T00645 CPG3A5 86302574 IC50 > 30000 nM T00645 C1HW4B 89735655 IC50 = 3000 nM T00645 C1E6PA 91938057 IC50 > 1000 nM T00645 CY7BI2 118706214 IC50 > 10000 nM T00645 CHT6K9 118728811 Ki > 4000 nM T00645 CUA3Y2 118728812 Ki > 4000 nM T00645 CDQ78G 118728813 Ki > 4000 nM T00645 CZ6XL7 118728814 Ki > 4000 nM T00645 CMO67K 118728815 Ki = 590 nM T00645 CR2M0Q 118728816 Ki > 4000 nM T00645 C62SCL 118728817 Ki > 4000 nM T00645 CSB30C 118728819 Ki = 490 nM T00645 CV7XU8 118728820 Ki = 230 nM T00645 C3J1EX 118728821 Ki > 4000 nM T00645 CIWB78 118728822 Ki > 4000 nM T00645 CP18SE 118728823 Ki > 4000 nM T00645 CM42CA 118728824 Ki = 1100 nM T00645 C9Q7CL 118728825 Ki > 4000 nM T00645 CCR3S0 118728826 Ki = 1500 nM T00645 CJQA40 122178640 Ki = 310 nM T00645 CK4Q1D 122178641 Ki = 500 nM T00645 CAW6X5 127047919 IC50 > 1000 nM T00645 C2AN7T 134611886 IC50 > 100000 nM T00645 CST7X3 135870706 IC50 < 50 nM T00645 CQ84IZ 136180335 Ki > 4000 nM T00645 D03DZO 11715767 IC50 > 10000 nM T00645 D05JRA 25190769 IC50 = 5.32 nM T00645 D07OXC 11650194 IC50 > 100000 nM T00645 D08HFG 24809764 IC50 > 10000 nM T00645 D0GT8N 5154691 IC50 = 500 nM T00645 D0T8NU 16757525 IC50 > 4000 nM T56510 D00PBX 49846579 Ki = 48 nM T56510 D02OZK 11404337 EC50 = 900 nM T56510 D06ETI 24978538 Ki = 0.055 nM T56510 D0I5DP 118910268 Ki = 700 nM T56510 D0U3EP 445154 IC50 = 190000 nM T56510 D0Z0HH 3503 Ki = 310 nM T56510 D03TTE 135513044 Ki = 420 nM T56510 D0B1UL 136002683 Ki = 240 nM T56510 D0CR9A 136183441 Ki = 370 nM T56510 D0L8WH 11228183 Ki < 0.5 nM T56510 D0R7MJ 135403797 IC50 = 2200 nM T56510 CJUW83 95696 Ki > 1000000 nM T56510 CMA78T 95864 Ki = 230000 nM T56510 CFMN24 234873 IC50 > 100000 nM T56510 C76CAZ 719016 Ki > 1000000 nM T56510 CMP56I 815185 Ki = 230000 nM T56510 C08YVK 819258 Ki > 1000000 nM T56510 CGAM30 1582605 Ki = 99000 nM T56510 CE48YZ 2729000 IC50 = 5100 nM T56510 CX8OI2 2797587 Ki = 500 nM T56510 CS5N4Q 3101542 Ki > 100000 nM T56510 CPS79F 3163284 Ki > 1000000 nM T56510 CTHP95 3951527 Ki = 4100 nM T56510 C1NX4W 3969372 Ki = 4700 nM T56510 CRP38E 4369509 Ki = 36 nM T56510 C3IUN5 5720188 Ki = 2400 nM T56510 C4A0NL 6436598 Ki > 100000 nM T56510 C3JX7W 6484626 Ki > 1000000 nM T56510 C3FIT9 6512895 IC50 = 3000 nM T56510 CE15GC 6519796 IC50 = 12600 nM T56510 CVBR15 6520864 IC50 = 17400 nM T56510 COG3E6 6535736 IC50 = 3400 nM T56510 C60XOG 10232933 Ki = 114 nM T56510 CWEL85 10792599 IC50 = 9500 nM T56510 C40IZU 11235484 Ki = 3313 nM T56510 CD40US 11246769 Ki = 1785 nM T56510 CA31FE 11316476 Ki = 781 nM T56510 CBL97Q 11339175 Ki = 5846 nM T56510 CL7R3U 11369024 IC50 = 2600 nM T56510 C0QDX2 11419664 Ki = 1013 nM T56510 CLET56 11459297 IC50 = 7400 nM T56510 C6N5MO 11463494 Ki = 10960 nM T56510 C6J7LA 11470999 IC50 > 100000 nM T56510 C62HQG 11471374 IC50 = 73000 nM T56510 C2VTX5 11498270 Ki = 471 nM T56510 CXK63W 11498475 Ki = 1.1 nM T56510 C1FO6C 11500877 IC50 = 625 nM T56510 CV4JK3 11502754 Ki = 75000 nM T56510 CVE4N6 11512578 IC50 > 50000 nM T56510 CJI08E 11512941 Ki = 665 nM T56510 C23QHG 11513027 Ki = 2.6 nM T56510 CU6KI5 11513202 Ki = 57.9 nM T56510 CQY3D8 11527399 Ki = 21.5 nM T56510 C7JYG1 11541153 Ki = 2520 nM T56510 CH6ZQ5 11541165 Ki = 1080 nM T56510 CKQ0Y7 11542308 Ki < 0.5 nM T56510 CMZ16P 11556440 Ki = 0.8 nM T56510 C6EIC4 11585288 Ki = 294 nM T56510 CATI96 11585498 Ki = 3.1 nM T56510 C3H1IL 11585607 Ki = 75 nM T56510 CI1U6J 11607072 Ki = 251 nM T56510 CRY85Q 11607405 Ki = 0.8 nM T56510 CZJL24 11610901 Ki = 1400 nM T56510 CZCQ84 11614246 Ki = 426 nM T56510 CNE9T7 11614353 Ki = 252 nM T56510 CJG0E3 11621908 Ki = 250 nM T56510 C6HB9W 11643296 Ki = 10.4 nM T56510 CPX8O4 11649997 Ki = 894 nM T56510 CJI48S 11650712 Ki = 1.7 nM T56510 CE3W8S 11657048 Ki = 19 nM T56510 C5SLF8 11657862 Ki < 0.5 nM T56510 C2O6HD 11679126 Ki = 38.9 nM T56510 CVL56F 11686025 Ki = 1 nM T56510 C0T9EK 11686478 Ki < 0.5 nM T56510 CJN6Y0 11700195 Ki = 396 nM T56510 CRIF42 11707282 Ki = 106 nM T56510 C3PY5U 11707606 Ki = 0.9 nM T56510 C9U7TI 11721651 Ki = 1.2 nM T56510 CZN62A 11750522 Ki = 839 nM T56510 C19DWM 11774143 Ki = 1852 nM T56510 CM7DS2 15991562 Ki = 0.8 nM T56510 C8IBM3 16109062 Ki = 4.6 nM T56510 CCSZ31 16109063 Ki = 1.3 nM T56510 C82PXV 16109064 Ki = 1.8 nM T56510 CD95NJ 16109065 Ki < 0.5 nM T56510 CRFU59 16109066 Ki = 0.9 nM T56510 CFQH70 16109067 Ki = 1.1 nM T56510 C07EWL 16109068 Ki < 0.5 nM T56510 CP1KE4 16109069 Ki = 0.9 nM T56510 CJ3ND2 16109076 Ki < 0.5 nM T56510 C15FQX 16109077 Ki < 0.5 nM T56510 COB84K 16109078 Ki < 0.5 nM T56510 C8NB6V 16109079 Ki = 0.6 nM T56510 C04ZCD 16109080 Ki < 0.5 nM T56510 CF9P2Y 16109081 Ki = 1.3 nM T56510 C4XDV1 16109084 Ki = 4.4 nM T56510 C5Q7XJ 16109088 Ki = 4 nM T56510 C6NWT1 16109089 Ki = 2.6 nM T56510 CVL8S5 16109090 Ki = 3 nM T56510 CUQ1N6 16109091 Ki < 0.5 nM T56510 CDHV39 16109092 Ki = 0.6 nM T56510 CXV9B1 16109093 Ki < 0.5 nM T56510 CMU3K7 16109094 Ki < 0.5 nM T56510 CN9EX7 16109095 Ki < 0.5 nM T56510 CXD2P4 16109096 Ki < 0.5 nM T56510 CX0G5D 16109097 Ki < 0.5 nM T56510 CW1R3F 16109098 Ki < 0.5 nM T56510 C6AX1T 16109099 Ki < 0.5 nM T56510 CUP40E 16109115 Ki = 3.7 nM T56510 C8TZ0R 16109116 Ki < 1 nM T56510 CF32ZY 16109117 Ki = 2.5 nM T56510 CHF2Y6 16109137 Ki = 6.1 nM T56510 C45VIE 16109138 Ki = 0.8 nM T56510 CJ65GB 16109139 Ki < 0.5 nM T56510 C6MKC4 16109140 Ki = 0.9 nM T56510 CT5R1N 16109141 Ki < 0.5 nM T56510 CSJ4A2 16109142 Ki < 0.5 nM T56510 CVS90W 16109149 Ki < 0.5 nM T56510 CT8Z1X 16109150 Ki < 0.5 nM T56510 CZ9OK8 16109151 Ki = 1.4 nM T56510 CD8C4M 16109152 Ki = 3.6 nM T56510 CR83BQ 16109153 Ki < 0.5 nM T56510 C5CTU8 16109154 Ki = 1.7 nM T56510 CKH97W 16109156 Ki < 0.5 nM T56510 C5NC8O 16109157 Ki = 0.9 nM T56510 C0QHV3 16109158 Ki < 0.5 nM T56510 CHP79I 16109159 Ki < 0.5 nM T56510 C6IZ8J 16109160 Ki < 0.5 nM T56510 CV8AB2 16109161 Ki < 0.5 nM T56510 C75YUM 16109162 Ki = 1 nM T56510 CI4Y5D 16109163 IC50 < 60 nM T56510 CV7HC8 16645886 Ki > 1000000 nM T56510 C06ZOQ 16681698 IC50 = 4690 nM T56510 C49JYU 22683787 Ki > 1000000 nM T56510 C7OZI2 24797083 IC50 > 80000 nM T56510 C5NI1B 24798804 IC50 = 3 nM T56510 CP18YW 25058454 IC50 = 26000 nM T56510 CMS0Z5 25058455 IC50 = 22000 nM T56510 C7GHE9 25099966 Ki > 10000 nM T56510 C4Z7CN 25100119 Ki > 15000 nM T56510 C74OSJ 25100590 Ki > 15000 nM T56510 C12LTS 25117879 IC50 = 64 nM T56510 CZ12DX 25229694 Ki = 190 nM T56510 CU34VF 25232834 IC50 = 13 nM T56510 CK78WE 42601456 Ki = 570 nM T56510 CHF9X2 42642427 Ki = 10800 nM T56510 CK21NB 44182311 IC50 = 11 nM T56510 CA9JF3 44191246 IC50 = 6300 nM T56510 C2FXA3 44191638 IC50 = 800 nM T56510 CXO2S9 44191694 IC50 = 800 nM T56510 CHT92S 44191696 IC50 = 930 nM T56510 C83UCJ 44191750 IC50 = 850 nM T56510 CMS39X 44191815 IC50 = 3500 nM T56510 C0J3RT 44192144 IC50 = 110 nM T56510 C97RQU 44192145 IC50 = 850 nM T56510 C57VCY 44224066 IC50 = 110 nM T56510 C5S0YV 44251267 Ki > 100000 nM T56510 C3N5SR 44278056 Ki > 30000 nM T56510 C4NH7R 44278214 Ki = 7631 nM T56510 CGM41H 44278239 Ki > 30000 nM T56510 CB3ZY6 44278271 Ki > 30000 nM T56510 C36SNO 44278284 Ki > 30000 nM T56510 CU2NP8 44278346 Ki > 30000 nM T56510 CJ5NV0 44278551 Ki = 10920 nM T56510 CP7O6U 44286285 Ki = 58900 nM T56510 C86DAF 44344017 IC50 = 180000 nM T56510 C06EXF 44344113 IC50 = 10000 nM T56510 CHK7U5 44473399 IC50 = 3000 nM T56510 CH95IX 44574943 Ki = 5700 nM T56510 CFD72X 44574944 Ki = 6600 nM T56510 CNO53W 44574945 Ki = 6000 nM T56510 C5YJF8 44574946 Ki = 11000 nM T56510 CH17BO 44574947 Ki = 5700 nM T56510 CHR74A 44574948 Ki = 7800 nM T56510 C68BOZ 44574949 Ki > 100000 nM T56510 C63BKT 44574950 Ki > 100000 nM T56510 CYD32H 44574951 Ki > 100000 nM T56510 CF6WN0 44574952 Ki > 100000 nM T56510 CNCZ86 44574953 Ki > 100000 nM T56510 CJTI53 44574954 Ki > 100000 nM T56510 CN02TB 44574955 Ki > 100000 nM T56510 CM45OJ 44574956 Ki > 100000 nM T56510 CQ9SA5 44574957 Ki > 100000 nM T56510 CH2E4R 44609307 Ki = 8050 nM T56510 C56ORH 44634480 Ki > 100000 nM T56510 C60ZXU 45140016 Ki = 3400 nM T56510 C9FUL6 45267264 Ki > 100000 nM T56510 C8OVQ7 45268131 Ki = 17800 nM T56510 C7WQ3U 45268134 Ki = 7600 nM T56510 CTM8C1 45269014 Ki = 7200 nM T56510 C4XM0N 45269015 Ki = 5300 nM T56510 CIU4T8 45269862 Ki > 100000 nM T56510 CR59JU 45269863 Ki > 100000 nM T56510 CHS2F0 45270488 Ki > 100000 nM T56510 CD0H5I 45270689 Ki > 100000 nM T56510 C3OG0N 46221373 IC50 = 12600 nM T56510 C7IT4V 46221374 IC50 = 6200 nM T56510 C0L6EQ 46221585 IC50 = 5200 nM T56510 C78ESU 46221586 IC50 = 1900 nM T56510 C8KZ3W 46221587 IC50 = 13400 nM T56510 CGF59X 46221588 IC50 = 35900 nM T56510 CYBC18 46221796 IC50 > 100000 nM T56510 CC6S8D 46222878 IC50 = 100000 nM T56510 CE38XU 46222879 IC50 = 12100 nM T56510 CWPA41 46222880 IC50 = 36000 nM T56510 C0EJ5G 46222881 IC50 = 12700 nM T56510 CF5PX1 46223098 IC50 = 26700 nM T56510 C4IGT6 46223099 IC50 = 5300 nM T56510 CZD7S3 46223100 IC50 = 10300 nM T56510 CBYX74 46223324 IC50 = 5400 nM T56510 CE2G5Z 46223325 IC50 = 19700 nM T56510 CIA79R 46223326 IC50 = 40400 nM T56510 C9D2TS 46223328 IC50 > 100000 nM T56510 C2IYE3 46223559 IC50 > 100000 nM T56510 CX3ZL6 46223560 IC50 > 100000 nM T56510 C07DWN 46223561 IC50 = 72000 nM T56510 CG2NH7 46236925 IC50 = 310 nM T56510 C78NZA 46236926 IC50 = 650 nM T56510 C3DV7L 46701726 Ki < 0.01 nM T56510 C4X8YH 46836110 IC50 = 7 nM T56510 C05NAZ 46836111 Ki = 5 nM T56510 CPDE67 46836168 Ki < 0.01 nM T56510 CF2ZB4 46836243 Ki = 12.4 nM T56510 CRG96F 46836244 Ki = 2.22 nM T56510 CY1XE2 46836305 Ki < 0.01 nM T56510 CY1E5M 46836567 IC50 = 91 nM T56510 CBM9P2 46836568 IC50 = 1 nM T56510 C9PG5S 46836648 IC50 = 86 nM T56510 C8ZHR7 46836862 Ki = 0.042 nM T56510 CSZT49 46837053 Ki = 0.34 nM T56510 CP1Y5L 46837056 IC50 = 270 nM T56510 C9TE5H 46842207 IC50 = 720 nM T56510 CZS89I 46887075 IC50 > 100000 nM T56510 CL18SN 46887149 IC50 = 6900 nM T56510 C9E3RI 46887150 IC50 = 7300 nM T56510 C4L8NR 46887151 IC50 > 100000 nM T56510 C3ZP0J 46887152 IC50 = 6200 nM T56510 CC8FB5 46907039 IC50 = 400000 nM T56510 C9P6KG 46907040 IC50 = 220000 nM T56510 CXW0L5 46907075 IC50 = 380000 nM T56510 C3PY8D 49840813 Ki = 8300 nM T56510 C74IAL 49846946 Ki = 14 nM T56510 CVBX71 51003001 IC50 = 650 nM T56510 CWQ69L 51003061 IC50 = 833 nM T56510 C8BZY6 51003123 IC50 = 291 nM T56510 C8IWO4 51346830 Ki = 127 nM T56510 CWK27M 51346831 Ki = 520 nM T56510 CSI02L 51346837 Ki = 170 nM T56510 C2ZT6I 51354614 IC50 = 34 nM T56510 C73DOP 51354615 IC50 = 6 nM T56510 CNA1W2 51354616 IC50 = 16 nM T56510 C4Q3YN 51354902 IC50 = 3 nM T56510 CON3Q1 51354903 IC50 = 20 nM T56510 C52OHD 51354904 IC50 = 3 nM T56510 CM3CU0 51355193 IC50 = 29 nM T56510 CZG7K2 52941339 EC50 = 579.43 nM T56510 CAK3Y7 52941340 EC50 = 100 nM T56510 CS5KO6 52941341 EC50 = 159.96 nM T56510 CM71WQ 52941342 EC50 = 389.94 nM T56510 C63TXD 52941343 EC50 = 799.83 nM T56510 CHX4F8 52941344 EC50 = 380.19 nM T56510 CNXF51 52941663 EC50 = 460.26 nM T56510 C7HP8F 52942558 EC50 = 380.19 nM T56510 C13TMQ 52942559 EC50 = 399.94 nM T56510 C1ME5A 52942560 EC50 = 149.97 nM T56510 C0IL5B 52942561 EC50 = 339.63 nM T56510 CIXL82 52942621 EC50 = 130.02 nM T56510 CXM25I 52942883 EC50 = 319.89 nM T56510 C0M9YO 52942884 EC50 = 34.99 nM T56510 C1XJ4C 52943761 EC50 = 749.89 nM T56510 CD89KL 52943762 EC50 = 230.14 nM T56510 CLX65M 52943763 EC50 = 149.97 nM T56510 CDCK18 52943764 EC50 = 149.97 nM T56510 CJUC36 52943765 EC50 = 1901.08 nM T56510 C71TGC 52944968 EC50 = 410.2 nM T56510 CX9M8H 52945020 EC50 = 55.98 nM T56510 C0MAB8 52945021 EC50 = 21.98 nM T56510 CV19GK 52945278 EC50 = 5495.41 nM T56510 CE9D3O 52946196 EC50 = 549.54 nM T56510 C92MLO 52946241 EC50 = 179.89 nM T56510 CNRP36 52946242 EC50 = 39.99 nM T56510 C3YAS0 52947426 EC50 = 1099.01 nM T56510 CXG6S9 52947427 EC50 = 17.99 nM T56510 CHN50K 52948645 EC50 = 680.77 nM T56510 C7K6MJ 52948646 EC50 = 250.03 nM T56510 CN7WK5 52948647 EC50 = 179.89 nM T56510 CHI3R6 52948648 EC50 = 619.44 nM T56510 CP1WU9 52948649 EC50 = 389.94 nM T56510 CW46YO 52948650 EC50 = 95.06 nM T56510 C15XBO 52948943 EC50 = 1099.01 nM T56510 C6UVC3 52949849 EC50 = 599.79 nM T56510 CZS32V 52949850 EC50 = 250.03 nM T56510 CBUD89 52949851 EC50 = 2600.16 nM T56510 C0T3WX 52949852 EC50 = 299.92 nM T56510 CU1FY0 52949853 EC50 = 660.69 nM T56510 CF03VA 52949897 EC50 = 29.99 nM T56510 CW9IN1 53234692 Ki = 630 nM T56510 CWTA43 53234693 Ki = 1710 nM T56510 CTPX94 53234694 Ki = 2080 nM T56510 CC34HU 53234695 Ki = 1940 nM T56510 CHL4C7 53234842 Ki = 1500 nM T56510 CZ8TK7 53234845 Ki = 1270 nM T56510 CS1ZG8 53235008 Ki = 16440 nM T56510 C6BA1V 53235009 Ki = 5820 nM T56510 CV75RW 53235092 Ki = 3420 nM T56510 C2K5GP 53235093 Ki = 6450 nM T56510 C9JD1C 53235169 Ki = 2290 nM T56510 C3Q9IV 53473132 IC50 = 9370 nM T56510 CD7O1T 53473133 IC50 = 3790 nM T56510 C4EW9Y 53473224 IC50 = 4140 nM T56510 CI9Z3T 53473225 IC50 = 28030 nM T56510 CK96PJ 53473226 IC50 = 33520 nM T56510 CD0T9X 53473227 IC50 = 49510 nM T56510 CCP0W5 53473228 IC50 = 161300 nM T56510 C98WGS 53473229 IC50 = 6200 nM T56510 C5T1HQ 53473314 IC50 = 310 nM T56510 CP9JX1 53473315 IC50 = 9980 nM T56510 C9QA7I 53473316 IC50 = 7150 nM T56510 CS5CP0 53473317 IC50 = 28520 nM T56510 C5M2UV 53473318 IC50 = 2530 nM T56510 CSZ78K 53473319 IC50 = 2310 nM T56510 C4HF7T 53473387 IC50 = 1940 nM T56510 CNVH01 53473388 IC50 = 1970 nM T56510 CU3J2D 53473389 IC50 = 4080 nM T56510 CCH9R0 53473390 IC50 > 1000000 nM T56510 CB2D9Z 53473391 IC50 = 10870 nM T56510 C78YZW 53473392 IC50 = 12110 nM T56510 C9Q0XS 53473478 IC50 = 2960 nM T56510 CX70AC 53473479 IC50 = 160 nM T56510 C6OTX3 53473480 IC50 = 3760 nM T56510 C1ME6Q 53473481 IC50 = 2700 nM T56510 CQHB31 53473482 IC50 = 2000 nM T56510 CHV0G1 53473570 IC50 = 2940 nM T56510 CN4O2V 53473571 IC50 = 2870 nM T56510 CSJ50X 53473572 IC50 = 86 nM T56510 C1O6KH 53473573 IC50 = 16770 nM T56510 C9L6JQ 53473574 IC50 = 15080 nM T56510 C9AYX8 53473660 IC50 = 42720 nM T56510 C1GY0B 53473661 IC50 = 3190 nM T56510 C50AOR 53473662 IC50 = 180 nM T56510 CU4RQ6 56933429 Ki < 1 nM T56510 CNKE09 56933430 IC50 = 7 nM T56510 CS3YP8 56933431 Ki < 1 nM T56510 C07IBG 56973535 IC50 = 47 nM T56510 CCN5O6 56973540 IC50 = 13 nM T56510 C9CEO1 57338853 IC50 = 394 nM T56510 C38QHP 57339126 Ki = 138000 nM T56510 CUK97J 57392876 Ki = 68 nM T56510 C1MQF6 57392877 Ki = 3.3 nM T56510 C38WES 57392878 Ki = 2.6 nM T56510 C5XN9L 57394832 Ki = 3910 nM T56510 C5XZ9E 57396359 Ki < 1 nM T56510 CSM8T4 57398377 Ki = 4840 nM T56510 CD0YR1 57403327 Ki = 1 nM T56510 CXP56B 57523339 Ki < 1 nM T56510 CX8EG1 57523340 Ki < 1 nM T56510 CC3KU7 57523369 Ki < 1 nM T56510 COA97D 57523370 Ki = 1.7 nM T56510 C61FYR 57523400 Ki < 1 nM T56510 CQ3L5W 57523401 Ki = 24.7 nM T56510 CH3I5T 57523430 Ki = 166000 nM T56510 C8P2QI 57523431 Ki = 5700 nM T56510 CX9BE7 57523432 Ki < 1 nM T56510 CF6IZ8 57523433 Ki < 1 nM T56510 C1YTI4 57523468 Ki = 8.3 nM T56510 C9AFI7 57523469 Ki = 1.7 nM T56510 C0OMZ9 57523470 Ki < 1 nM T56510 C4RDZ5 57523498 Ki < 1 nM T56510 C5LM1Z 58531411 IC50 > 30000 nM T56510 CRN79Z 59053435 IC50 = 14 nM T56510 CHM9V8 59053436 IC50 = 5 nM T56510 C6Y1KZ 59053563 IC50 = 32 nM T56510 CNFW46 59053624 Ki < 1 nM T56510 CJHN01 59053688 IC50 = 26 nM T56510 CL8B3J 59053755 IC50 = 8.3 nM T56510 C40SFQ 59053932 IC50 = 9.4 nM T56510 CIR74F 59438327 IC50 = 20 nM T56510 C04ELI 59447491 Ki = 0.04 nM T56510 CW1MT4 59447501 Ki = 0.03 nM T56510 CQF73L 59447527 Ki = 0.02 nM T56510 C1OX3J 59447540 IC50 = 16 nM T56510 CYK9T2 59447570 Ki = 0.01 nM T56510 CUE6O3 59447571 IC50 = 4 nM T56510 CBLR64 59447577 Ki < 0.01 nM T56510 CH9XY2 59447590 IC50 = 90 nM T56510 C51EJI 59447629 IC50 = 610 nM T56510 CBW6X9 59447631 IC50 = 32 nM T56510 C7E0NU 59447641 IC50 = 43 nM T56510 C52IXR 60169703 Ki < 1 nM T56510 CN28ME 60169704 Ki < 1 nM T56510 CI13RU 60169705 Ki = 1.2 nM T56510 C49HLF 60169795 Ki < 1 nM T56510 CHAV90 60169796 Ki < 1 nM T56510 CI93MH 60171063 Ki = 88000 nM T56510 C3GRZ0 60204010 Ki < 1 nM T56510 CZPD50 66561644 IC50 = 44 nM T56510 CUVL40 66561645 IC50 = 12 nM T56510 CQ8MS0 66561714 IC50 = 10 nM T56510 CR2Y5X 66561715 IC50 = 14 nM T56510 C0DV3M 66561716 IC50 = 9 nM T56510 CT5X6W 68453674 IC50 = 150 nM T56510 C3GH9F 70495544 IC50 = 4.7 nM T56510 CZM1G2 70495760 IC50 = 5.9 nM T56510 CUM37L 70496039 IC50 = 6.1 nM T56510 C2W5BS 70680244 Ki > 15000 nM T56510 CF5OC7 70680245 Ki > 15000 nM T56510 C34TMX 70681580 IC50 = 30 nM T56510 CG53LQ 70681581 IC50 = 35 nM T56510 C85SWT 70681582 IC50 = 140 nM T56510 CK5G2S 70681583 IC50 = 480 nM T56510 CT92UD 70681589 IC50 = 150 nM T56510 CGO1Z2 70681590 IC50 = 47 nM T56510 CBWI18 70683696 IC50 = 18 nM T56510 CV01CQ 70683697 IC50 = 15 nM T56510 C5ZGR4 70683707 IC50 = 130 nM T56510 C4R9SX 70683708 IC50 = 16 nM T56510 C1FAS8 70683709 IC50 = 26 nM T56510 CJ3YR9 70684416 Ki < 1 nM T56510 C5QD1R 70685844 IC50 = 470 nM T56510 CR4CN7 70685853 IC50 = 970 nM T56510 CCFR15 70685854 IC50 = 37 nM T56510 CTYS31 70686561 Ki = 11.3 nM T56510 C76YLJ 70687968 IC50 = 640 nM T56510 CM4L9Q 70687969 IC50 = 26 nM T56510 CL5ZN3 70687970 IC50 = 120 nM T56510 CCN32L 70687971 IC50 = 500 nM T56510 CJR4L6 70687978 IC50 = 710 nM T56510 C2A8PT 70689990 IC50 = 11 nM T56510 CC4E1T 70689991 IC50 = 48 nM T56510 CK26AI 70689992 IC50 = 55 nM T56510 CJK6O0 70689993 IC50 = 15 nM T56510 C0AL5K 70690001 IC50 = 160 nM T56510 C7WQ1I 70690002 IC50 = 230 nM T56510 COI13D 70690003 IC50 = 4300 nM T56510 C7ERL2 70690004 IC50 = 23 nM T56510 CHW46I 70690005 IC50 = 590 nM T56510 CF43BG 70692160 IC50 = 41 nM T56510 CACR07 70692161 IC50 = 54 nM T56510 C2WX0B 70692162 IC50 = 17 nM T56510 CFO0R7 70692163 IC50 = 17 nM T56510 CG10VQ 70692164 IC50 = 29 nM T56510 CRAI92 70694200 IC50 = 42 nM T56510 C4OFB8 70694201 IC50 = 35 nM T56510 CG6Z3T 70694202 IC50 = 13 nM T56510 C16TJP 70694203 IC50 = 6 nM T56510 CWBC96 70694204 IC50 = 7 nM T56510 CY4B1M 70694205 IC50 = 7 nM T56510 C38ZQO 70694215 IC50 = 120 nM T56510 CAN0R1 70694216 IC50 = 24 nM T56510 CIJX30 70694217 IC50 = 22 nM T56510 CMO3U8 70694218 IC50 = 19 nM T56510 C7VY3B 70696312 IC50 = 8 nM T56510 CR56GE 70696317 IC50 = 250 nM T56510 CI4DG1 70696318 IC50 = 550 nM T56510 CY39FW 70696319 IC50 = 62 nM T56510 CL3W0R 71297203 IC50 = 1.5 nM T56510 CH3TN5 71297204 IC50 = 13 nM T56510 CRV98Q 71297207 Ki = 1.1 nM T56510 CF58GV 71297208 IC50 = 500 nM T56510 C8C7FS 71451698 EC50 = 6200 nM T56510 CE03NH 71453306 Ki < 1 nM T56510 CJA8N4 71455243 EC50 > 100000 nM T56510 COH24E 71455246 EC50 > 100000 nM T56510 CVC5F8 71455247 EC50 > 100000 nM T56510 CUG8N7 71462421 EC50 = 14600 nM T56510 CVF0O2 71545164 Ki = 15000 nM T56510 C4E1FO 71545167 Ki > 15000 nM T56510 CAW6K1 71545330 Ki > 15000 nM T56510 CHPJ72 71545486 Ki > 15000 nM T56510 CS92IM 71545651 Ki > 15000 nM T56510 CC7I6A 71545824 Ki = 6800 nM T56510 CGL67T 71545826 Ki > 15000 nM T56510 CBW68J 71545828 Ki > 15000 nM T56510 CS14HM 71545993 Ki = 4100 nM T56510 C0HP4B 71545994 Ki = 6800 nM T56510 CP3Y2O 71548702 Ki = 9590 nM T56510 CS02CG 71549001 Ki = 15140 nM T56510 C37AJW 71549412 Ki = 48150 nM T56510 C3LIN4 71565985 Ki < 0.01 nM T56510 CTH79R 71605747 IC50 = 15 nM T56510 CZ4BU0 71605927 IC50 = 12 nM T56510 CG8Z1K 71605928 IC50 = 13 nM T56510 CAZ2N3 71605929 IC50 = 4.5 nM T56510 CY7L5E 71606084 IC50 = 6 nM T56510 C6UVA9 71606085 IC50 = 4.7 nM T56510 CR3ZA7 71606086 IC50 = 18 nM T56510 C7XK8P 71606257 IC50 = 15 nM T56510 C9G6DT 71606258 IC50 = 5 nM T56510 C6K8BA 71606424 IC50 = 8.2 nM T56510 CK1C8L 71606584 IC50 = 16 nM T56510 CJX1Y4 71624427 IC50 = 24 nM T56510 CW3QY0 71654876 Ki = 520 nM T56510 CU6X2Z 71656178 Ki = 5540 nM T56510 CCI0N7 71656179 Ki > 660 nM T56510 CYFW14 71716172 IC50 = 22 nM T56510 C9WS6R 71716944 IC50 = 74 nM T56510 C1ZDP3 71717609 Ki = 21 nM T56510 C53RPU 71718227 Ki = 500 nM T56510 CW4DP2 71719220 IC50 = 20 nM T56510 CNH94Q 71719979 IC50 = 115 nM T56510 CVQ6G2 71720436 IC50 = 62 nM T56510 CR7ZV1 71747665 IC50 > 100000 nM T56510 CKM8N3 71747851 IC50 = 2000 nM T56510 CDSK62 72672102 IC50 = 6 nM T56510 C16WOR 72715983 IC50 = 22000 nM T56510 CE84VA 72715984 IC50 = 13000 nM T56510 CRM08G 72793103 IC50 > 30000 nM T56510 C6C8FO 72793104 IC50 = 8000 nM T56510 CX86EJ 72793174 IC50 = 150 nM T56510 CY23TP 72793175 IC50 = 7.2 nM T56510 CS5R9Y 72793176 IC50 = 4.4 nM T56510 CB6E4W 72793245 IC50 = 3.7 nM T56510 CO6E8W 73213478 Ki = 8700 nM T56510 CDO87T 73213545 Ki = 1200 nM T56510 C9G8FB 73213546 Ki = 2100 nM T56510 C90NSV 73214548 Ki = 2200 nM T56510 C0TAJ1 73334912 Ki = 90 nM T56510 CNF20H 73345953 IC50 = 14 nM T56510 C9D8CK 73347484 IC50 = 10 nM T56510 C3WBM5 73347485 IC50 = 47 nM T56510 C7O1BG 73347486 IC50 = 41 nM T56510 CVC6Z1 73349009 IC50 = 49 nM T56510 CI7P6T 73349010 IC50 = 17 nM T56510 CNU9I6 73349011 IC50 = 100 nM T56510 C6KWN5 73349012 IC50 = 77 nM T56510 CDB2C3 73350570 IC50 = 51 nM T56510 C4VS5K 73350571 IC50 = 78 nM T56510 C2KIX7 73352077 IC50 = 55 nM T56510 C6ZGJ8 73353547 IC50 = 20 nM T56510 CK4B3L 73355044 IC50 = 60 nM T56510 CJ8MA1 73355661 IC50 > 40000 nM T56510 CW35TO 73356596 IC50 = 130 nM T56510 CWCB85 73356597 IC50 = 260 nM T56510 C3C7QO 86765310 Ki = 10580 nM T56510 C04RXD 90316425 IC50 > 100000 nM T56510 CMC8E7 90478312 Ki > 100000 nM T56510 CF06DQ 90478313 Ki = 3400 nM T56510 CZ7T8W 90478318 Ki = 3100 nM T56510 CEK6S7 90478319 Ki = 2400 nM T56510 CMP47T 90478320 Ki = 6800 nM T56510 CX6WP8 90644931 IC50 > 20000 nM T56510 CV59BT 90644932 IC50 = 1000 nM T56510 CF09DY 90644933 IC50 = 9200 nM T56510 C5HE1T 90644934 IC50 = 9600 nM T56510 CBL0J2 90644935 IC50 = 5300 nM T56510 C7IM5P 90644936 IC50 = 5100 nM T56510 CX0D2H 90644937 IC50 > 100000 nM T56510 C6Y1GD 90645494 Ki > 100000 nM T56510 CV0AI7 90645495 Ki = 19200 nM T56510 CP06VM 90645496 Ki = 12600 nM T56510 CN24WU 90645497 Ki > 100000 nM T56510 CU8G4Y 90645498 Ki = 19400 nM T56510 CFSJ09 90645499 Ki > 100000 nM T56510 C79THC 90656473 Ki > 15000 nM T56510 C12JEQ 91754241 Ki > 20000 nM T56510 C20WCK 102360805 Ki = 150 nM T56510 CHL0X1 118394626 Ki > 40000 nM T56510 CO40GK 118394721 Ki > 40000 nM T56510 CE28ZO 118394843 Ki > 40000 nM T56510 C3BQH4 118394951 Ki > 40000 nM T56510 CQT5W4 118406840 Ki > 36000 nM T56510 CY1L9S 118406932 Ki = 11000 nM T56510 CBTM73 118406950 Ki > 36000 nM T56510 CA7DW1 118406955 Ki = 19000 nM T56510 CEOY82 118406960 Ki > 36000 nM T56510 CW4K9Y 118406985 Ki > 36000 nM T56510 CPN23M 118406995 Ki > 36000 nM T56510 CR4K9M 118705735 IC50 = 15 nM T56510 C2Q7JN 118705736 IC50 = 25 nM T56510 C23NUF 118705737 IC50 = 38 nM T56510 C27WRY 118705738 IC50 = 10 nM T56510 CT09UA 118705739 IC50 = 10 nM T56510 CN6T8R 118705740 IC50 = 10 nM T56510 CA6X5L 118705741 IC50 = 33 nM T56510 C9I0TA 118705742 IC50 = 138 nM T56510 C5G7LA 118707175 IC50 = 63 nM T56510 CD3K7L 118707176 IC50 > 1000 nM T56510 C2R8UD 118707281 IC50 = 378 nM T56510 C37IQC 118707282 IC50 = 39 nM T56510 CKN64C 118707283 IC50 = 98 nM T56510 CR1Y9J 118707284 IC50 = 77 nM T56510 CP70CG 118707285 IC50 = 308 nM T56510 CJ9D4H 118707286 IC50 = 18 nM T56510 CI7D3R 118707287 IC50 = 38 nM T56510 CU0ZT2 118707288 IC50 < 10 nM T56510 CF4LD2 118707289 IC50 = 31 nM T56510 C6LV2K 118707290 IC50 = 11 nM T56510 COU9T1 118707291 IC50 = 54 nM T56510 CTX75Y 118707292 IC50 = 21 nM T56510 C1LD3P 118707293 IC50 < 10 nM T56510 CI5OV2 118707294 IC50 < 10 nM T56510 CO1GM8 118707295 IC50 = 30 nM T56510 C6FM7I 118707296 IC50 < 10 nM T56510 CFG28Y 118707297 IC50 = 21 nM T56510 C8JGF6 118723013 Ki = 9000 nM T56510 C1LD6S 118727814 Ki = 930 nM T56510 CLGO34 118727815 Ki = 17 nM T56510 CGK28A 118727816 Ki = 4100 nM T56510 CI7C8K 118727817 Ki = 1100 nM T56510 CY5U7E 118728671 Ki = 520 nM T56510 C4BDN6 118728672 Ki = 730 nM T56510 C6O0NI 118728673 Ki = 2400 nM T56510 CZ9AW7 118728674 Ki = 630 nM T56510 CWOB25 118728675 Ki = 410 nM T56510 CVB3L2 118728676 Ki = 950 nM T56510 C5YE4D 118728677 Ki = 460 nM T56510 CJ0EA7 118728678 Ki = 460 nM T56510 CSE54F 118728679 Ki = 420 nM T56510 C1QW4O 118728680 Ki = 470 nM T56510 CG81OQ 118728681 Ki = 470 nM T56510 C23OKP 118728682 Ki = 540 nM T56510 C1L2WK 118728683 Ki = 450 nM T56510 C6HIF9 118728684 Ki = 510 nM T56510 CX2V0P 118728685 Ki = 540 nM T56510 CR4SL3 118728686 Ki = 1900 nM T56510 CBVR49 118728687 Ki = 2400 nM T56510 CUA45V 118728688 Ki = 660 nM T56510 C14VIN 118728689 Ki = 1400 nM T56510 CK32FL 118728690 Ki = 800 nM T56510 CFUB67 118728691 Ki = 870 nM T56510 C4OG6B 118728692 Ki = 850 nM T56510 C1MXB4 118728693 Ki = 50000 nM T56510 C1B6PH 118728694 Ki = 700 nM T56510 C8XBN6 118728695 Ki = 710 nM T56510 C37NXV 118728696 Ki = 360 nM T56510 C9WX0R 118728697 Ki = 1200 nM T56510 CO25VC 118728698 Ki = 900 nM T56510 C30CAD 118728699 Ki = 5600 nM T56510 C40UFD 118728700 Ki = 750 nM T56510 CUY95K 118728701 Ki = 680 nM T56510 C95MPZ 118728702 Ki = 750 nM T56510 CVR7L2 118728703 Ki = 720 nM T56510 CG24YU 118728704 Ki = 80 nM T56510 CM2B9A 118734788 Ki > 100000 nM T56510 CF73NP 118734789 Ki > 100000 nM T56510 C5W2EA 118734957 Ki > 660 nM T56510 CU5S7Y 118737140 Ki = 9000 nM T56510 CO5K1H 118737141 Ki > 20000 nM T56510 C8HLR2 118737142 Ki = 12700 nM T56510 C40BQS 118737143 Ki > 20000 nM T56510 C9BJR5 118737144 Ki = 1900 nM T56510 C4G0TJ 118737145 Ki > 20000 nM T56510 CNW6B0 118737146 Ki = 7400 nM T56510 CLV10W 118737147 Ki > 20000 nM T56510 CW29QH 118737148 Ki > 20000 nM T56510 CRE89M 118737149 Ki = 3000 nM T56510 C51KLE 118737150 Ki = 4700 nM T56510 C0EA6G 118737151 Ki > 20000 nM T56510 CPS8Z2 118737152 Ki > 20000 nM T56510 CQ8M7Y 118737153 Ki > 20000 nM T56510 C1ERH8 118737154 Ki = 7800 nM T56510 CN7ZE6 118737156 Ki > 20000 nM T56510 CP9MA5 118737157 Ki = 5200 nM T56510 C2FOD3 118737158 Ki > 20000 nM T56510 CUX2N7 122193137 Ki = 3900 nM T56510 CDJE95 122193145 Ki > 10000 nM T56510 C5S6PU 122193146 Ki > 10000 nM T56510 CA0KR9 122194475 Ki = 6100 nM T56510 C4ODZ9 122194476 Ki > 50000 nM T56510 CXTI31 122194478 Ki > 50000 nM T56510 CM7Y4S 122194479 Ki = 4700 nM T56510 CA45FG 122194480 Ki > 50000 nM T56510 C9SRV7 122194632 Ki > 10000 nM T56510 CUI60T 122194634 Ki > 10000 nM T56510 CNK8M7 122194635 Ki > 10000 nM T56510 CR19KU 122622656 Ki > 25000 nM T56510 CE4MG7 122622800 Ki > 25000 nM T56510 CBFO10 122622827 Ki = 6600 nM T56510 CY9OL2 122623097 Ki = 5200 nM T56510 C1R4UJ 122633925 Ki > 25000 nM T56510 C03SVJ 127031331 Ki = 1566 nM T56510 CHQY05 127031601 Ki > 50000 nM T56510 C38FBK 127031602 Ki > 50000 nM T56510 CIG1C9 127031603 Ki = 4467 nM T56510 COW3X7 127031604 Ki = 1109 nM T56510 CCU25Z 127031889 Ki = 943 nM T56510 C3UQ5T 127031890 Ki = 997 nM T56510 CW2DY9 127032749 Ki = 4467 nM T56510 C5JI4W 127033064 Ki = 12854 nM T56510 CER6M1 127033065 Ki > 50000 nM T56510 CWY3K5 127033066 Ki = 1404 nM T56510 CJZT46 127033067 Ki = 9069 nM T56510 CJ2G6T 127033347 Ki > 50000 nM T56510 C2EU0Y 127036597 Ki = 2 nM T56510 CIBD06 127044491 Ki = 2500 nM T56510 C7KGI0 127044661 Ki = 8400 nM T56510 CAY7Q9 127050688 Ki = 17 nM T56510 C81IYU 134131766 Ki = 160 nM T56510 CBZ96D 134133726 Ki = 140 nM T56510 CJ7RT9 134135886 Ki = 290 nM T56510 C0MAL5 134137174 Ki = 70 nM T56510 C1D4WS 134137526 Ki > 20000 nM T56510 C91HZY 134139104 Ki = 120 nM T56510 C9ME1S 134140038 Ki > 20000 nM T56510 CM0X8W 134141608 Ki = 110 nM T56510 CSFE39 134144182 Ki = 130 nM T56510 C0SLU6 134148123 Ki = 330 nM T56510 C1UHN8 134151998 Ki = 1300 nM T56510 C2VC8J 134152063 Ki = 450 nM T56510 C7ZH8I 134152922 Ki = 210 nM T56510 CW4EP2 134153984 Ki = 320 nM T56510 C9ATX6 134154502 Ki = 170 nM T56510 CQ24RE 134154949 Ki = 210 nM T56510 CZ9Q5K 134155175 Ki = 290 nM T56510 C61URW 134155768 Ki = 510 nM T56510 CFG1Z7 134157505 Ki = 90 nM T56510 C2INR6 134828256 Ki > 40000 nM T56510 CSDR07 135157296 IC50 > 1000 nM T56510 CL98UM 135340006 Ki = 135000 nM T56510 CY1SE5 135691163 IC50 > 50000 nM T56510 C9MFV2 136002682 Ki = 160 nM T56510 C6FY0E 136002684 Ki = 210 nM T56510 CU0YE2 136032534 Ki = 2000 nM T56510 CASH13 136032535 Ki = 8400 nM T56510 C9RD0X 136032611 Ki = 110 nM T56510 CC09EN 136183442 Ki = 2070 nM T56510 CYJD84 136183443 Ki = 960 nM T56510 CF8HV7 136183446 IC50 = 76 nM T56510 C9TM5X 136190478 IC50 = 171 nM T56510 C1P6OX 136190479 IC50 = 43 nM T56510 C7QX1I 136190480 IC50 = 37 nM T56510 C6DTX1 136217518 IC50 = 85 nM T56510 CQ76AY 136217524 IC50 = 165 nM T56510 C1BOF5 136217525 IC50 = 71 nM T56510 CAB04U 136217526 IC50 = 18 nM T56510 CO86YC 136217527 IC50 = 315 nM T56510 C2GM7B 136217528 IC50 = 181 nM T56510 C6P5FM 136217530 IC50 = 283 nM T56510 CO40EL 136217531 IC50 = 162 nM T56510 C1EY2P 136229638 IC50 > 50000 nM T56510 CCG19P 136252244 IC50 = 53 nM T56510 CDG12L 136252252 Ki = 4690 nM T56510 C7GNK8 136259626 IC50 = 6 nM T56510 C7IRN8 136934823 Ki > 100000 nM T56510 CG25KR 136934824 Ki > 100000 nM T56510 C6OG0P 136934825 Ki = 30900 nM T56510 CN07GX 136934826 Ki > 100000 nM T56510 C8Z4PU 136934827 Ki > 100000 nM T56510 C1W4YP 136934828 Ki = 15500 nM T56510 CS6Z1D 136934829 Ki > 100000 nM T56510 CE9O5J 136934830 Ki = 3400 nM T56510 CLP4D9 137631972 Ki = 26000 nM T56510 CFU98I 137634219 Ki = 6200 nM T56510 CKF09I 137634986 Ki = 21000 nM T56510 CTX58M 137641044 Ki = 710 nM T56510 CGA35P 137641809 Ki > 36000 nM T56510 CBY3S6 137644084 Ki = 2100 nM T56510 CX9A0P 137654155 Ki > 36000 nM T56510 C1G3HA 141721113 Ki = 25000 nM T56510 CJ24FY 141721128 Ki > 40000 nM T56510 CS5M3A 141721326 Ki = 26000 nM T56510 CY0S1E 145946042 EC50 > 31500 nM T56510 C89JBL 145949373 Ki > 23000 nM T56510 C1RH9D 145950508 Ki = 15630 nM T56510 C3Y2MT 145950725 Ki > 23000 nM T56510 C01PGN 145951197 Ki > 23000 nM T56510 CG1U0T 145951885 Ki = 2730 nM T56510 C4JY1B 145951938 Ki = 14080 nM T56510 C13BLU 145952150 Ki > 23000 nM T56510 CJ9RW7 145952398 Ki = 5310 nM T56510 CMP86N 145952997 Ki > 23000 nM T56510 CR86NC 145953250 Ki = 2190 nM T56510 CDRT57 145953525 Ki = 8480 nM T56510 C15HUW 145953591 Ki > 23000 nM T56510 C8VIT4 145954556 Ki = 20730 nM T56510 CKM98O 145954557 Ki > 23000 nM T56510 C6C9UX 145955049 Ki = 9910 nM T56510 C3YPX4 145955393 Ki = 480 nM T56510 CT32ER 145955454 Ki > 23000 nM T56510 C0DFZ5 145956250 Ki = 3920 nM T56510 CXA7J4 145956350 Ki > 23000 nM T56510 CPWL30 145956560 Ki > 23000 nM T56510 CQ56PE 145956913 Ki > 23000 nM T56510 C5VPR7 145957258 Ki > 23000 nM T56510 CTLC26 145958175 Ki = 840 nM T56510 C6ZH2C 145958475 Ki = 510 nM T56510 CDJL71 145958776 Ki > 23000 nM T56510 CH23LV 145958880 Ki > 23000 nM T56510 C40QTV 145959015 Ki > 23000 nM T56510 CC82IQ 145959586 Ki = 16470 nM T56510 CBEH81 145964348 IC50 = 105 nM T56510 CL7K3I 145965147 IC50 = 59.3 nM T56510 CB7G6P 145965660 IC50 = 116 nM T56510 CG7P1Z 145966192 IC50 = 26.6 nM T56510 C2RJ4H 145966654 IC50 = 218 nM T56510 C5SN3Q 145966763 IC50 > 1000 nM T56510 CNSQ67 145967322 IC50 = 55.3 nM T56510 C3XRD8 145967779 IC50 = 29.3 nM T56510 C5FL7B 145968700 IC50 > 1000 nM T56510 CB5O9E 145971233 Ki = 2740 nM T56510 CH51QR 145972482 Ki = 2440 nM T56510 CGAZ83 145972946 Ki = 4400 nM T56510 C7R5ED 145973286 IC50 = 14.6 nM T56510 C37LPJ 145973505 IC50 = 13.2 nM T56510 CYQR17 145973714 IC50 = 25.6 nM T56510 CU65EX 145974322 Ki = 1910 nM T56510 CM6U1R 145976325 IC50 > 1000 nM T56510 CD8Q9R 145976379 IC50 = 162 nM T56510 C52PKW 145977421 IC50 = 49.3 nM T56510 C2QPU1 145977736 IC50 = 342 nM T56510 C9LBE6 145978364 IC50 = 33.5 nM T56510 CL76CK 145978956 IC50 = 765 nM T56510 CKF3S0 145979166 IC50 = 970 nM T56510 CGIZ51 145979582 IC50 > 1000 nM T56510 CZUD98 145979683 IC50 = 287 nM T56510 CL0H3M 145979783 IC50 = 270 nM T56510 C0NJC3 145982309 IC50 > 1000 nM T56510 CP39XU 145985660 IC50 = 109 nM T56510 CI6K3W 145986491 IC50 = 71.9 nM T56510 CU9I4K 145989784 IC50 > 1000 nM T56510 C7WT5C 145989980 IC50 > 1000 nM T56510 CSZ4M5 145990737 IC50 = 279 nM T56510 CTVC87 145991099 IC50 > 1000 nM T56510 CQ8M0P 145991800 IC50 = 512 nM T56510 C4BM9U 145991913 IC50 > 1000 nM T56510 C2OG0L 145993372 IC50 > 1000 nM T56510 C9KI8G 145993554 IC50 > 1000 nM T56510 C0NWC7 145993811 IC50 = 624 nM T56510 CW4O5A 145993860 IC50 > 1000 nM T56510 CCVP03 145994390 Ki > 25000 nM T56510 C78QAT 155513044 EC50 > 31500 nM T56510 C9Z8FQ 155514893 Ki = 216000 nM T56510 CTE3V7 155515598 Ki = 26000 nM T56510 CJ7A1D 155516576 Ki = 42000 nM T56510 CB37YD 155518816 IC50 = 1060 nM T56510 CLP32K 155519706 Ki = 287000 nM T56510 CUJY40 155521076 Ki = 18000 nM T56510 C3HYI9 155524558 Ki = 319000 nM T56510 CN1U6Q 155524659 Ki = 87000 nM T56510 C6W9LH 155524710 Ki = 17000 nM T56510 CXY0L3 155527670 Ki = 15000 nM T56510 C8WGO3 155530396 EC50 > 31500 nM T56510 C4ZNJ7 155534814 Ki = 107000 nM T56510 CV3L8Q 155536071 Ki = 18000 nM T56510 CNAR96 155536134 EC50 = 5630 nM T56510 CK7UQ4 155537237 IC50 = 50 nM T56510 CEAJ80 155539156 Ki = 24000 nM T56510 C8CEJ5 155542773 Ki = 39000 nM T56510 CUS28M 155542793 Ki = 3500 nM T56510 C6TQ4X 155545656 EC50 = 2420 nM T56510 CL4HF7 155547093 Ki = 6700 nM T56510 C7E9FH 155554727 IC50 = 4.6 nM T56510 CUX0F2 155558443 IC50 = 350 nM T56510 CYIB91 155563107 Ki = 33000 nM T56510 C5Y0QF 155565915 EC50 = 4080 nM T56510 C8CL3Z 155569283 EC50 = 2380 nM T56510 CWOV84 44580965 IC50 = 5000 nM T56510 CF8B9I 59053554 Ki = 1500 nM T56510 CN10OD 59053562 IC50 = 22 nM T56510 D00LHS 11455910 Ki = 1110 nM T56510 D05RDP 992586 Ki = 7850 nM T56510 D0D6BH 379493 IC50 = 8500 nM T56510 D0G2JZ 1464 Ki = 0.9 nM T56510 D0T3VP 2782689 EC50 > 31500 nM T56510 D0V7PX 454878 IC50 = 1700 nM T58921 D00WCX 39042 EC50 = 3000 nM T58921 D05DVP 5717 EC50 = 2440 nM T58921 D05LYX 3488 Ki = 660 nM T58921 D05VIX 3463 EC50 = 147800 nM T58921 D07XGR 3339 EC50 = 570 nM T58921 D0G2MW 446284 IC50 = 1600 nM T58921 D0J5DC 2796 EC50 = 500000 nM T58921 D0K5ER 5281055 Ki = 14 nM T58921 D0N6RF 65999 EC50 = 700 nM T58921 D0NF1U 64929 IC50 > 10000 nM T58921 D0O1TC 5280581 IC50 = 2400 nM T58921 D0R1RS 3715 EC50 = 50000 nM T58921 D0UE9X 5280933 IC50 = 2200 nM T58921 D00AUX 25230266 EC50 = 961 nM T58921 D00PJJ 9869229 EC50 = 163 nM T58921 D00SWQ 10429242 EC50 = 657 nM T58921 D02NHD 447458 Ki = 90 nM T58921 D03OSG 11236126 EC50 > 1000 nM T58921 D04BPS 9888484 IC50 = 33.96 nM T58921 D04QIE 11526038 EC50 = 1100 nM T58921 D06QBY 10229498 EC50 = 4 nM T58921 D08PFA 3055168 EC50 = 43 nM T58921 D09DJC 9863341 EC50 = 8.6 nM T58921 D0AX9S 446642 EC50 = 0.2 nM T58921 D0H1NL 208901 EC50 = 13 nM T58921 D0I5IM 135449333 IC50 = 6500 nM T58921 D0LW1Y 9864881 EC50 = 2116 nM T58921 D0M0SS 170364 EC50 = 0.3388 nM T58921 D0M3UT 206044 EC50 = 3 nM T58921 D0U0KR 3035850 Ki = 2.18 nM T58921 D0VU5M 9890879 EC50 = 4 nM T58921 D0X7VB 12082259 EC50 > 500 nM T58921 D0Y8NZ 9832447 EC50 = 0.038 nM T58921 D0H5FI 9958543 EC50 = 1 nM T58921 D0PO7F 10143056 EC50 = 2 nM T58921 D00YGA 9845965 EC50 = 1 nM T58921 D05HDX 9803963 EC50 = 800 nM T58921 D08LZI 9947731 EC50 = 6850 nM T58921 D0B0EB 9890585 EC50 = 3.981 nM T58921 D0B8JQ 9825046 EC50 = 2500 nM T58921 D0B9EN 10274777 IC50 = 19 nM T58921 D0GS7N 183134 EC50 > 20000 nM T58921 D0YO4D 3922 EC50 = 18.6 nM T58921 C9RN3W 7127 EC50 = 40000 nM T58921 CSB8Q0 8215 IC50 = 30000 nM T58921 CVT2C4 10467 IC50 = 30000 nM T58921 CX3V5T 33584 IC50 = 40000 nM T58921 CZ8B2Q 60560 EC50 = 7600 nM T58921 CQ3H6U 60910 IC50 = 140000 nM T58921 C1GZ6P 128814 IC50 > 10000 nM T58921 C80LUR 154005 EC50 = 3940 nM T58921 C3O9HN 286310 EC50 = 15.3 nM T58921 CUC68S 339720 EC50 > 10000 nM T58921 C0SBX4 431161 EC50 = 224 nM T58921 CU89CQ 441964 Ki = 54000 nM T58921 C3VPB4 445655 IC50 = 30 nM T58921 C20GQD 446758 EC50 = 169.82 nM T58921 C12SCN 637584 EC50 = 58600 nM T58921 C2FE3L 643734 EC50 = 16700 nM T58921 C85OXQ 725701 EC50 = 2511.89 nM T58921 CZN6S9 743974 IC50 > 25118.86 nM T58921 C3KWX2 1020637 EC50 = 215 nM T58921 CX8B2V 1201193 IC50 = 876 nM T58921 C3RU4T 1209375 IC50 = 1144 nM T58921 C17AOB 1231560 IC50 = 7970 nM T58921 CTF16Y 1284989 EC50 = 2290 nM T58921 C9KP6J 1285388 IC50 = 20000 nM T58921 CX6H1A 1389211 IC50 = 5132 nM T58921 C4F7DS 1543988 IC50 = 1319 nM T58921 C5ZN1R 1551564 IC50 = 1326 nM T58921 CTY13X 2280142 EC50 = 9000 nM T58921 CB2X0E 2285412 EC50 = 8000 nM T58921 CFV29H 2287582 EC50 = 10000 nM T58921 C8VO6N 2742752 IC50 = 512 nM T58921 C8G4QW 2742758 IC50 = 175 nM T58921 CGL1J4 2742759 EC50 = 0.78 nM T58921 C5D7YX 2745807 EC50 = 2100 nM T58921 C75IAD 2746797 EC50 = 5400 nM T58921 CLU85B 2772717 IC50 = 2223 nM T58921 CEO3V6 2772783 Ki = 3715.35 nM T58921 CJX4U2 2800607 EC50 = 200 nM T58921 CP5OT3 2805771 EC50 = 600 nM T58921 COE0Y8 2813539 EC50 = 3100 nM T58921 CIZ40Y 2813684 EC50 = 2800 nM T58921 C7TFW2 2851123 IC50 = 100 nM T58921 CRF26V 2892191 EC50 = 3300 nM T58921 C38KAD 2892375 EC50 = 10000 nM T58921 C6M3KG 3114052 EC50 > 10000 nM T58921 C8LJS6 3114053 EC50 = 4800 nM T58921 CMPX57 3114054 EC50 = 3600 nM T58921 C8AG4S 3114055 EC50 = 8600 nM T58921 CG38HZ 3114056 EC50 = 9300 nM T58921 C8QGD7 3584988 IC50 = 26000 nM T58921 CCU6W0 3820637 Ki = 7100 nM T58921 C3F2QR 4147757 EC50 = 680 nM T58921 COH6I9 4287647 EC50 = 1600 nM T58921 CT29VZ 4388708 EC50 = 682 nM T58921 C32LKN 4518233 IC50 = 40000 nM T58921 CH34WN 5281116 IC50 = 30000 nM T58921 C6K2GJ 5281805 EC50 = 26940 nM T58921 CQAJ80 5289162 EC50 = 1300 nM T58921 C75ORQ 5310669 EC50 = 15380 nM T58921 CX98HV 5312835 EC50 > 20 ug.mL-1 T58921 C72UVI 5319482 Ki = 18100 nM T58921 CJ8P4T 5352624 EC50 = 800 nM T58921 CH7Z5F 5534504 EC50 = 7000 nM T58921 CZ0D2P 5715241 EC50 = 22290 nM T58921 CZ6T5I 5829359 IC50 = 382 nM T58921 CT0F3V 5863774 IC50 = 747 nM T58921 CY4CO5 5889656 IC50 = 302 nM T58921 CG37TN 5967793 IC50 = 2098 nM T58921 CDV7S3 5975420 IC50 = 1439 nM T58921 C73ABY 6027581 IC50 = 703 nM T58921 CUEK97 6036014 IC50 = 1294 nM T58921 CCR25A 6058603 IC50 = 1088 nM T58921 CZJ84H 6102812 IC50 = 50 nM T58921 CC6L1G 6161619 IC50 = 407 nM T58921 C83MFH 6241863 IC50 = 10712 nM T58921 CK8E3N 6270191 IC50 = 1187 nM T58921 CM3LK8 6300697 IC50 = 13521 nM T58921 C16ZSG 6439929 IC50 = 27000 nM T58921 C1VU9T 6440462 IC50 = 850 nM T58921 CLO7Y1 6540257 IC50 = 210 nM T58921 CJDX25 7009663 IC50 = 8670 nM T58921 C4P2OK 7135379 EC50 = 15000 nM T58921 CGXH64 9547900 IC50 = 152 nM T58921 CM85OW 9549238 IC50 = 3 nM T58921 C50PDQ 9549255 EC50 > 10000 nM T58921 CF6VL8 9796107 Ki = 3890.45 nM T58921 C3CXT4 9802192 EC50 = 30 nM T58921 C5PGB8 9803821 EC50 = 800 nM T58921 C7TMX8 9805639 IC50 = 22 nM T58921 CCMF21 9806390 EC50 = 12000 nM T58921 C9R7OA 9822722 Ki = 52 nM T58921 CQK19U 9822766 EC50 = 400 nM T58921 C47ZRD 9823501 EC50 = 7040 nM T58921 C7DP5Y 9824628 EC50 = 16700 nM T58921 CXB52G 9825302 EC50 = 1500 nM T58921 C8WSD7 9825400 Ki = 30 nM T58921 CSY86D 9825523 IC50 > 15000 nM T58921 CJF2M6 9826186 EC50 = 500 nM T58921 CZ9MW3 9839556 EC50 = 33800 nM T58921 CD04KR 9844059 EC50 = 490 nM T58921 CR7J1B 9844286 EC50 = 9800 nM T58921 CSZ36U 9844554 EC50 = 1500 nM T58921 CRA1O5 9844638 EC50 = 57 nM T58921 C7Z4YA 9845640 EC50 = 750 nM T58921 C0Z2DQ 9845736 EC50 = 2400 nM T58921 C9RM5A 9845832 EC50 = 4200 nM T58921 CQ1ZH6 9847065 EC50 = 7.4 nM T58921 CP5MW0 9847836 EC50 = 200 nM T58921 C6ABL9 9850395 EC50 = 2400 nM T58921 CS5DU2 9863468 Ki = 147.91 nM T58921 C7S3YF 9866595 EC50 = 4.677 nM T58921 CD4RY0 9867298 EC50 = 760 nM T58921 C70MKO 9868387 EC50 = 3700 nM T58921 CAE0R3 9868664 EC50 = 12.2 nM T58921 CX7C0D 9868836 EC50 = 1700 nM T58921 C7VLA1 9869022 EC50 = 1200 nM T58921 CRC51S 9869157 EC50 = 2.7 nM T58921 CWJU60 9870703 EC50 = 26300 nM T58921 CJ3AD7 9888213 EC50 = 4000 nM T58921 C90UXQ 9889347 EC50 = 6.4 nM T58921 C7CB6G 9893080 IC50 = 490 nM T58921 C6O1SV 9895808 EC50 = 4 nM T58921 CY9O3C 9902264 EC50 = 1100 nM T58921 C0NI1K 9908951 EC50 = 12100 nM T58921 C1BIG0 9910452 EC50 = 12600 nM T58921 CTW75H 9910503 EC50 = 117 nM T58921 C57LHY 9910951 IC50 = 46 nM T58921 C0A3UZ 9911319 EC50 = 1.3 nM T58921 C57EPL 9931070 EC50 = 91 nM T58921 CM7I8Y 9931437 EC50 = 100 nM T58921 C1G6FX 9932058 EC50 = 6400 nM T58921 C75NOF 9932563 EC50 = 2700 nM T58921 C9PCJ5 9932790 EC50 = 1610 nM T58921 CH32AQ 9933395 EC50 = 8250 nM T58921 CGV83S 9933541 EC50 = 2700 nM T58921 CF7P8W 9934050 EC50 = 7300 nM T58921 C4VKF5 9934858 EC50 = 3790 nM T58921 C8OQX3 9935996 EC50 = 1210 nM T58921 CWVJ56 9949411 EC50 = 10000 nM T58921 CH5EF9 9955171 EC50 = 760 nM T58921 CH4S2G 9955206 EC50 = 3400 nM T58921 C2VHT3 9955922 EC50 > 3000 nM T58921 CRE2W1 9956726 EC50 = 9700 nM T58921 C02YNS 9956737 EC50 = 160 nM T58921 C5R9BK 9959189 EC50 = 67 nM T58921 CQP9I8 9960726 EC50 = 1650 nM T58921 CV74OZ 9980586 IC50 = 24 nM T58921 C45OEJ 9980930 IC50 > 15000 nM T58921 CFKD10 9981617 EC50 > 3000 nM T58921 CF0SR7 9982519 EC50 = 9 nM T58921 CJOV70 9983904 EC50 = 20 nM T58921 C0GBI5 9985365 EC50 = 23 nM T58921 CH7W9P 10003213 EC50 = 3630780.55 nM T58921 CM1BQ5 10003577 EC50 = 0.4 nM T58921 CKJ83Z 10004270 EC50 = 3 nM T58921 C8JV7T 10004390 Ki = 30 nM T58921 CIZJ14 10005136 IC50 > 50000 nM T58921 C6VP7J 10005230 IC50 = 6770 nM T58921 CK24FM 10005763 EC50 = 4677351.41 nM T58921 C6C9SG 10005877 EC50 = 710 nM T58921 CID1R9 10021239 IC50 = 50 nM T58921 C0OED7 10023279 EC50 = 1100 nM T58921 C64EJL 10027350 IC50 = 5400 nM T58921 CLK7R6 10028864 IC50 = 450 nM T58921 CZEI65 10043645 Ki = 1949.84 nM T58921 C6LG4U 10044126 EC50 = 700 nM T58921 C7KI8V 10047627 IC50 > 10000 nM T58921 CQH15A 10053715 EC50 > 10000 nM T58921 CBS0U5 10068664 EC50 = 43.65 nM T58921 C48JGT 10070650 EC50 = 990 nM T58921 CNS96V 10072967 IC50 = 15 nM T58921 CCG14W 10073789 EC50 = 20 nM T58921 CJRY94 10074505 EC50 = 20417379.45 nM T58921 CC72JH 10074964 EC50 = 58884365.54 nM T58921 C79TZB 10075037 EC50 = 4265795.19 nM T58921 CO2IN7 10075041 EC50 = 29512092.27 nM T58921 C9PH1M 10075336 EC50 = 18197008.59 nM T58921 CR01QE 10076802 EC50 = 100 nM T58921 CL53DC 10091852 EC50 = 883 nM T58921 CM5EU7 10093355 EC50 = 2000 nM T58921 C3ZT0K 10096907 IC50 = 8000 nM T58921 CQ2EH0 10096908 EC50 = 160 nM T58921 CRJU50 10098103 EC50 = 32 nM T58921 C8BWY7 10109101 EC50 = 30000 nM T58921 CK6Y4X 10112293 EC50 = 100 nM T58921 CI5E6O 10112797 EC50 = 46 nM T58921 CZU39A 10113515 EC50 = 239 nM T58921 C94TCV 10113516 EC50 = 3800 nM T58921 CW5KR2 10113686 IC50 > 15000 nM T58921 CQG9E4 10113721 EC50 = 820 nM T58921 CWH2U3 10113980 IC50 = 1698.24 nM T58921 CL7TY9 10114135 EC50 = 294 nM T58921 C1BA8V 10114442 EC50 = 700 nM T58921 C6FIV9 10115344 IC50 = 43.95 nM T58921 C1EOY3 10116365 IC50 = 2700 nM T58921 C15GVJ 10116451 EC50 = 1600 nM T58921 C7ROV3 10116541 IC50 = 2140 nM T58921 C8UQ9G 10116787 EC50 = 20 nM T58921 CY73BR 10117908 EC50 > 10000 nM T58921 CTGB91 10118056 IC50 = 370 nM T58921 CRCG14 10118927 Ki = 420 nM T58921 CM56XR 10119125 EC50 = 2 nM T58921 CFZ80V 10119392 EC50 = 7 nM T58921 C98ENV 10119393 EC50 = 6 nM T58921 CU89OW 10119824 EC50 = 4 nM T58921 CWGV68 10136347 EC50 = 136 nM T58921 C74VJE 10136660 IC50 = 13 nM T58921 C8O0AV 10137115 EC50 = 61 nM T58921 C2N6UZ 10137230 EC50 = 3900 nM T58921 CDX37J 10137693 EC50 = 500 nM T58921 CVI26N 10138146 EC50 > 10000 nM T58921 CMRP39 10139247 EC50 = 8 nM T58921 CB3SH2 10139551 EC50 = 19 nM T58921 C6RPI1 10139836 EC50 = 1000 nM T58921 C6N1TJ 10140233 EC50 = 400 nM T58921 CBE62A 10140247 EC50 = 21 nM T58921 CS53BZ 10141294 IC50 = 914 nM T58921 CR4E1D 10141305 EC50 > 10000 nM T58921 CB53WS 10141607 IC50 = 3 nM T58921 C0OD9X 10141609 EC50 = 13000 nM T58921 CQM84R 10142329 EC50 = 124 nM T58921 C78OLG 10143678 EC50 = 19 nM T58921 CW04MX 10144243 EC50 = 2 nM T58921 CIXB29 10157662 EC50 = 212 nM T58921 CKH28L 10157940 EC50 = 35 nM T58921 CAMN64 10158648 EC50 = 274 nM T58921 C7XT5K 10159635 EC50 > 10000 nM T58921 C4XM1D 10160128 EC50 = 42 nM T58921 CYB95E 10161728 EC50 = 534 nM T58921 C05LIH 10161760 EC50 = 16 nM T58921 C4T7GE 10161854 Ki = 38 nM T58921 C95FYK 10161996 EC50 = 12 nM T58921 C9C3JQ 10162008 IC50 = 520 nM T58921 CZ24HT 10162063 EC50 = 800 nM T58921 C7DU6F 10162210 EC50 = 360 nM T58921 CDM26O 10162519 EC50 = 3000 nM T58921 CMF69H 10162615 EC50 = 2500 nM T58921 C6JB5Q 10162929 EC50 = 290 nM T58921 C6AE1Y 10163556 EC50 > 10000 nM T58921 CFE2M9 10163810 IC50 = 2200 nM T58921 CZ6EW0 10164032 EC50 = 1800 nM T58921 CM21IJ 10164033 EC50 = 4000 nM T58921 C9FR3O 10174350 IC50 = 23600 nM T58921 C2RL8N 10177074 IC50 = 2760 nM T58921 C93CIF 10177377 Ki = 1120 nM T58921 C5JHK0 10181314 EC50 = 32 nM T58921 C52QCT 10182727 EC50 = 16 nM T58921 CDT75W 10182946 EC50 = 700 nM T58921 C7I1LS 10183245 EC50 = 77 nM T58921 CUQ89L 10183490 IC50 = 6194.41 nM T58921 C49HSN 10183977 IC50 > 15000 nM T58921 CO93AD 10184159 EC50 = 19 nM T58921 CRUV90 10184204 EC50 = 540 nM T58921 CJ0ER3 10184971 EC50 = 12 nM T58921 C7V1ML 10186118 EC50 = 168 nM T58921 CFCY37 10186986 Ki = 1.479 nM T58921 CDF82U 10199589 EC50 = 27 nM T58921 CPM13H 10201545 EC50 = 2000 nM T58921 CVD5N1 10202000 EC50 = 15 nM T58921 C7NPZ3 10202354 Ki = 365 nM T58921 CJ0R3W 10202547 EC50 = 4 nM T58921 C1J2VR 10204076 EC50 = 6 nM T58921 CC3G0I 10204762 EC50 = 1000 nM T58921 CYA5S6 10204908 EC50 = 3000 nM T58921 CFD6Z2 10205060 EC50 = 191 nM T58921 CY1ZK2 10205220 EC50 = 8 nM T58921 C0F5CK 10205615 EC50 = 205 nM T58921 CAQ5U8 10205828 IC50 = 1700 nM T58921 CZ7A6O 10206788 EC50 = 160 nM T58921 CMSG62 10207241 EC50 = 170 nM T58921 C6MYJ4 10207242 EC50 = 5000 nM T58921 CM4HS7 10207244 EC50 = 1400 nM T58921 CO52SH 10208214 IC50 = 630 nM T58921 CL4R0K 10208548 EC50 = 3 nM T58921 C03WGI 10208599 Ki = 47 nM T58921 C1NIA4 10217191 IC50 > 10000 nM T58921 CPAH95 10222749 EC50 = 73 nM T58921 CL1K2N 10223023 IC50 = 20.99 nM T58921 C9VEU1 10223369 EC50 = 13 nM T58921 C9SIT0 10223583 EC50 = 228 nM T58921 CI57ZX 10223837 EC50 = 34 nM T58921 CS25KJ 10224123 EC50 = 59 nM T58921 CY28GC 10224783 EC50 = 1200 nM T58921 C4R7LT 10224945 EC50 = 1 nM T58921 CQ56VG 10225637 EC50 = 600 nM T58921 CU1T0A 10225684 EC50 = 22 nM T58921 CJH81C 10225731 EC50 = 10000 nM T58921 C2RY6K 10225793 EC50 = 14 nM T58921 CYR3B5 10226233 EC50 = 260 nM T58921 CG4P7X 10226511 EC50 = 3000 nM T58921 CVAT07 10226701 IC50 = 84 nM T58921 C7U0ZQ 10226739 EC50 = 120 nM T58921 CUS8V5 10227653 IC50 = 10000 nM T58921 CSL75P 10228304 EC50 = 19 nM T58921 CS7Q9U 10229225 EC50 = 750 nM T58921 C8J0AZ 10230642 EC50 = 50 nM T58921 COVB68 10252612 EC50 = 760 nM T58921 CC8GU0 10254028 EC50 = 15488166.19 nM T58921 CARH74 10254209 EC50 = 470 nM T58921 C2HIT7 10254845 IC50 = 399 nM T58921 C3OE5Z 10257392 EC50 = 40 nM T58921 CDX58E 10257647 IC50 = 109 nM T58921 C9KZJ3 10270710 IC50 = 1200 nM T58921 CTBJ17 10273040 EC50 = 1200 nM T58921 CVH34N 10274499 EC50 = 40 nM T58921 C4PM2S 10274627 EC50 = 10000 nM T58921 CR6L1U 10274642 EC50 = 45 nM T58921 CH59WA 10274664 EC50 = 5 nM T58921 CJCU12 10274955 EC50 = 206 nM T58921 CZ64AI 10275334 EC50 > 10000 nM T58921 C72YHL 10275376 EC50 = 5400 nM T58921 C73ZHW 10276052 Ki = 110 nM T58921 CI1BV7 10276470 EC50 = 2800 nM T58921 C7YMO1 10276539 Ki = 3 nM T58921 C2KZ4D 10277333 EC50 = 14 nM T58921 CIOK04 10277666 EC50 = 160 nM T58921 C02EHS 10279905 IC50 = 1 nM T58921 CW34DF 10280116 EC50 = 730 nM T58921 CSJ28C 10280496 IC50 = 3 nM T58921 CS1U0K 10281422 EC50 = 2800 nM T58921 CW9HU6 10288123 EC50 = 5 nM T58921 CCN93S 10294697 EC50 = 42 nM T58921 C6JO3D 10295984 EC50 = 260 nM T58921 CQR18V 10295993 EC50 > 10000 nM T58921 CY28SU 10296059 EC50 = 3900 nM T58921 CP2MO0 10296330 EC50 = 1900 nM T58921 CK7F1O 10297427 EC50 = 1000 nM T58921 CO1P5R 10297760 IC50 = 13 nM T58921 CL40QG 10297943 EC50 > 10000 nM T58921 CXA6K2 10298514 EC50 = 670 nM T58921 CLE54O 10298859 EC50 = 104 nM T58921 CL5WB3 10299983 EC50 = 400 nM T58921 CS9V4N 10300072 EC50 = 3600 nM T58921 C89QXN 10300073 EC50 = 1200 nM T58921 CVP6R4 10300190 EC50 = 30 nM T58921 C7UNX1 10300279 EC50 > 10000 nM T58921 CLQD46 10301814 EC50 = 670 nM T58921 CFS25Z 10320822 EC50 = 140 nM T58921 CQH6P7 10323352 EC50 = 10715193.05 nM T58921 CDU6H7 10323599 EC50 = 22908676.53 nM T58921 C7S4LC 10324316 EC50 = 10 nM T58921 CTZ42X 10337211 Ki = 221.4 nM T58921 CGD4N7 10341169 EC50 = 280 nM T58921 C01MTP 10341401 EC50 = 530 nM T58921 CG58VR 10341444 EC50 > 15000 nM T58921 C46JQA 10341445 EC50 = 14000 nM T58921 C6HM5O 10342769 EC50 = 190 nM T58921 C8AT6R 10342801 EC50 > 3000 nM T58921 C3NJ4S 10343538 EC50 = 120 nM T58921 CB6R4D 10344769 EC50 = 70 nM T58921 CPO38A 10345547 EC50 = 540 nM T58921 C92PZC 10346786 EC50 = 30 nM T58921 CPT82D 10347115 EC50 = 50118723.36 nM T58921 CR5P7Z 10347250 IC50 = 210 nM T58921 C0OP5K 10347566 IC50 = 20 nM T58921 C0HOY8 10356158 EC50 = 400 nM T58921 COR01K 10363179 EC50 = 4800 nM T58921 C23JXU 10367018 EC50 > 3000 nM T58921 C0SKH9 10368050 IC50 = 3110 nM T58921 CMW4U5 10368444 EC50 = 12022644.35 nM T58921 CDA5F7 10369999 IC50 = 40 nM T58921 CB8KU1 10370056 IC50 = 90 nM T58921 CC1IK3 10370262 EC50 > 10000 nM T58921 COX30V 10371027 IC50 = 1 nM T58921 C0SLF7 10371709 EC50 = 110 nM T58921 CN92GI 10387634 EC50 = 4 nM T58921 C8LG4Z 10390333 EC50 = 300 nM T58921 CJQV19 10391684 EC50 = 90 nM T58921 C7PO5N 10392711 Ki = 1.413 nM T58921 C4GD0W 10408561 EC50 = 690 nM T58921 CTMS40 10409008 EC50 = 6480 nM T58921 CQY70C 10409988 IC50 = 196 nM T58921 C9GLW7 10410878 EC50 = 3 nM T58921 C29PFI 10412116 EC50 = 10 nM T58921 C5AWB0 10414708 EC50 = 56 nM T58921 CBN4H0 10415698 EC50 = 60 nM T58921 CND0P9 10431756 EC50 = 310 nM T58921 C72JHZ 10432356 EC50 = 770 nM T58921 CTQ0R7 10433053 EC50 = 1100 nM T58921 CKGE28 10434749 EC50 = 3235936.57 nM T58921 CU8Z4B 10437965 IC50 = 33 nM T58921 C4PFX2 10438226 EC50 = 3 nM T58921 C63QBA 10455509 EC50 = 90 nM T58921 CWQ2K1 10455511 IC50 = 38 nM T58921 CT7PM6 10455681 EC50 = 3311311.21 nM T58921 C1S7GU 10455871 EC50 = 3388441.56 nM T58921 C4DXE1 10457843 EC50 = 8709635.9 nM T58921 C1H5RP 10458842 EC50 = 85113803.82 nM T58921 C05UYW 10460941 EC50 = 1.288 nM T58921 C9Q5HV 10480558 EC50 = 60 nM T58921 CJ6S2A 10480923 EC50 = 24547089.16 nM T58921 CP04MX 10481007 EC50 = 5754399.37 nM T58921 CGXY36 10482372 EC50 = 4 nM T58921 CX8WS4 10493001 Ki = 14900 nM T58921 CQWS73 10506648 Ki = 2.344 nM T58921 CLUP75 10506906 Ki = 33.11 nM T58921 CY31MB 10506909 EC50 = 15.14 nM T58921 CL69EZ 10507132 EC50 = 0.1 nM T58921 CFE67K 10527748 Ki = 794.33 nM T58921 CXW3T7 10528164 Ki = 977.24 nM T58921 CES31O 10528836 Ki = 112.2 nM T58921 C18OWD 10528951 Ki = 18.62 nM T58921 CL86MF 10529251 Ki = 794.33 nM T58921 C2LVU0 10530201 Ki = 158.49 nM T58921 CE8Z9M 10530998 Ki = 1.738 nM T58921 CR1O9Z 10531248 EC50 = 0.6026 nM T58921 C5QUJ6 10550530 EC50 = 691.83 nM T58921 CK3L1A 10553219 Ki = 537.03 nM T58921 CP5A8D 10553649 Ki = 549.54 nM T58921 C9GJD6 10554575 EC50 = 1.072 nM T58921 CJ2O0B 10554759 EC50 = 51.29 nM T58921 C04RCN 10554988 EC50 = 1.047 nM T58921 CIHV75 10577962 Ki = 3.715 nM T58921 C8IJ2O 10578273 Ki = 32.36 nM T58921 CU8QT4 10578478 Ki = 2.57 nM T58921 CT1CU8 10578561 Ki = 162.18 nM T58921 CMPY58 10578809 EC50 = 5.012 nM T58921 CY4F5V 10578925 Ki = 0.8913 nM T58921 CXY5I4 10579996 Ki = 66.07 nM T58921 C4CM0Q 10597892 EC50 = 489.78 nM T58921 CAPK07 10600977 Ki < 3162.28 nM T58921 CHLZ07 10601672 Ki = 371.54 nM T58921 CGFO01 10602101 Ki = 107.15 nM T58921 C1B8PZ 10602637 Ki = 0.6918 nM T58921 C4LGB3 10624045 Ki = 371.54 nM T58921 C5MID1 10624243 Ki = 51.29 nM T58921 CWDF95 10624526 Ki = 1380.38 nM T58921 C07NWZ 10625055 Ki = 93.33 nM T58921 C6Q7HC 10625172 Ki = 15.49 nM T58921 CSDW83 10626484 Ki = 1380.38 nM T58921 CZG3C2 10626761 Ki = 0.871 nM T58921 CSV7L1 10626890 Ki = 123.03 nM T58921 C9H1UT 10627009 Ki = 416.87 nM T58921 CR1TO0 10627213 Ki = 42.66 nM T58921 CQ0J7E 10627451 Ki = 2.63 nM T58921 CWL48D 10648401 Ki = 1023.29 nM T58921 C7UR1G 10648889 Ki = 6.457 nM T58921 C38OBD 10649454 Ki = 251.19 nM T58921 CYX2C6 10649715 Ki = 234.42 nM T58921 CS07RU 10650300 Ki = 2.239 nM T58921 CGN6E1 10650503 Ki = 467.74 nM T58921 C04XGH 10673872 Ki = 132739445.8 nM T58921 C3I6CF 10674028 EC50 = 2.884 nM T58921 CS49NP 10674186 Ki = 1445.44 nM T58921 C6GV9A 10674474 EC50 = 0.1259 nM T58921 CMTU60 10674509 EC50 = 0.2455 nM T58921 CET39D 10674573 Ki = 8.71 nM T58921 CBL6H3 10674589 Ki = 4.365 nM T58921 CFY8L0 10695518 Ki = 354.81 nM T58921 CZ29WD 10696048 Ki = 269.15 nM T58921 C3V6NS 10696530 Ki = 1023.29 nM T58921 CA1QP6 10697014 Ki = 724.44 nM T58921 CU9D4M 10697739 Ki = 1548.82 nM T58921 CR2TL4 10697795 Ki = 676.08 nM T58921 C1SWC6 10698099 Ki = 19.5 nM T58921 C4PIH1 10698305 Ki = 0.7762 nM T58921 C63WVI 10698507 Ki = 1621.81 nM T58921 C3K8FY 10698557 EC50 = 2.692 nM T58921 CM05KO 10698874 Ki = 5.129 nM T58921 CPZG21 10721272 Ki = 1.259 nM T58921 CXH30Z 10721362 Ki = 13.49 nM T58921 CX6N0C 10721363 Ki = 3.311 nM T58921 C26MKN 10723133 Ki = 0.9772 nM T58921 C8KNR9 10743135 EC50 = 6 nM T58921 CVF19J 10743777 Ki = 104.71 nM T58921 CB8UJ5 10743977 Ki = 9.333 nM T58921 CCQ6R0 10744911 Ki = 154.88 nM T58921 CX8DT5 10745039 Ki = 23.44 nM T58921 C74DPN 10745235 Ki = 2.692 nM T58921 CB8DN9 10745789 Ki = 5.248 nM T58921 CC03DH 10746194 Ki = 2.692 nM T58921 CQ86RI 10746316 EC50 = 23.99 nM T58921 C07ANU 10746810 Ki = 2.63 nM T58921 CE05VH 10767544 Ki = 346.74 nM T58921 CZ69VT 10767943 Ki = 117.49 nM T58921 CF12XM 10768484 Ki = 6.457 nM T58921 CF7W9N 10769067 EC50 = 0.2818 nM T58921 CGI0V4 10792302 Ki = 27.54 nM T58921 CYE68O 10792674 Ki = 4.786 nM T58921 CJCM42 10792741 Ki = 2.818 nM T58921 CSA48Q 10793321 Ki = 954.99 nM T58921 CGF14Z 10793522 Ki = 1.995 nM T58921 C08EAW 10811786 Ki = 11.75 nM T58921 C41UAH 10814547 Ki = 128.82 nM T58921 C0X2GS 10814768 Ki = 38.9 nM T58921 C1KEY6 10815148 Ki = 131.83 nM T58921 CA4N5P 10816129 Ki = 85.11 nM T58921 CMDZ08 10816473 Ki = 1174.9 nM T58921 CK73BF 10816799 Ki = 72.44 nM T58921 CO38EU 10839028 Ki = 2398.83 nM T58921 CKM3B7 10839878 Ki = 91.2 nM T58921 CNMX53 10840119 Ki = 758.58 nM T58921 CL41RI 10840202 Ki = 2.754 nM T58921 CEQV19 10840203 EC50 = 3.467 nM T58921 CD8YV4 10840507 EC50 = 7.762 nM T58921 CP9J3U 10840584 Ki = 2.57 nM T58921 C3QZM9 10840711 Ki = 2.291 nM T58921 CK6F4C 10840712 Ki = 5.623 nM T58921 CZG96J 10896097 EC50 > 50000 nM T58921 CFW9J2 10896153 EC50 = 330 nM T58921 C5J4PX 10896495 EC50 > 50000 nM T58921 CYI87W 10914801 EC50 = 10000 nM T58921 C6UIW4 10983398 EC50 = 1716 nM T58921 C80VSA 10992201 EC50 = 2751 nM T58921 C5BN4L 11024616 IC50 = 10591 nM T58921 CJBM20 11042473 EC50 = 19300 nM T58921 CF38JZ 11048469 EC50 = 2800 nM T58921 CRK95E 11049998 EC50 = 43.65 nM T58921 CSJ7R0 11058026 EC50 = 2059 nM T58921 CG23SM 11071056 EC50 > 50000 nM T58921 C8E4YR 11133305 EC50 = 7400 nM T58921 C5KB7N 11153268 IC50 = 3160 nM T58921 C61TQH 11154732 EC50 > 1000 nM T58921 CM1RV7 11154887 EC50 = 264 nM T58921 CQ13LJ 11155087 IC50 = 35 nM T58921 CG2V4U 11155122 EC50 = 669 nM T58921 CIV54T 11155356 EC50 > 1000 nM T58921 C3LG4F 11155783 EC50 = 20 nM T58921 CP9NX6 11156185 EC50 = 2600 nM T58921 CN47MW 11165712 EC50 = 12 nM T58921 CLA09R 11165781 IC50 = 2980 nM T58921 CN7QF3 11166818 EC50 = 50 nM T58921 CIW98T 11167613 EC50 = 25 nM T58921 CF0H2Q 11167738 EC50 = 69 nM T58921 C3OWD7 11169884 EC50 = 320 nM T58921 CQE3O5 11176532 EC50 ~ 5000 nM T58921 CSO27I 11177525 IC50 = 4680 nM T58921 C4W7XI 11178006 EC50 = 182 nM T58921 C6IZ7D 11178075 IC50 = 210 nM T58921 CJR25A 11178155 EC50 = 300 nM T58921 C1M9TC 11178156 EC50 = 120 nM T58921 CW2FH7 11178750 EC50 = 1 nM T58921 CM3BO2 11178916 EC50 = 285 nM T58921 C6BQ7O 11179502 EC50 = 30 nM T58921 CY3LO2 11184855 EC50 = 19952.62 nM T58921 C01XFA 11186225 EC50 = 8900 nM T58921 C3EGQ4 11186282 IC50 = 1220 nM T58921 C30RIO 11187864 EC50 > 5000 nM T58921 CXA72P 11188236 EC50 = 197 nM T58921 CK84AR 11188766 IC50 > 10000 nM T58921 C50QOG 11189474 IC50 = 85 nM T58921 C8EIV0 11189652 EC50 = 360 nM T58921 C2D9FS 11190667 EC50 = 30 nM T58921 CA7K4Q 11190685 EC50 > 1000 nM T58921 C7B0QN 11190733 EC50 = 1000 nM T58921 CQ42YC 11199906 EC50 = 13 nM T58921 C89UCH 11202658 IC50 = 440 nM T58921 C2JK4F 11203145 EC50 = 900 nM T58921 CYHZ54 11208735 EC50 = 18860 nM T58921 C7ZPE1 11211156 EC50 > 1000 nM T58921 C71NVH 11211999 EC50 = 156 nM T58921 C9Z2HY 11212004 EC50 = 208 nM T58921 CO73VY 11212480 IC50 = 200 nM T58921 CU2F0D 11213609 EC50 = 2.9 nM T58921 C7P2LF 11214000 EC50 = 1981 nM T58921 C3G7FR 11214539 EC50 > 3000 nM T58921 CM6I2B 11218775 EC50 = 7200 nM T58921 C1Y8BI 11221515 EC50 > 5000 nM T58921 C4X5YO 11222878 EC50 > 5000 nM T58921 C7S9CH 11223211 IC50 = 210 nM T58921 C92VLZ 11223613 IC50 = 75 nM T58921 C8ZH4J 11224385 EC50 = 2700 nM T58921 C8JZ6Q 11225048 EC50 = 8 nM T58921 C8ATL5 11225797 EC50 = 898 nM T58921 CJ78RY 11225851 EC50 > 3000 nM T58921 CE4I3N 11225910 EC50 > 1000 nM T58921 CD2NX7 11227195 EC50 > 25000 nM T58921 CQJ5E6 11234410 EC50 = 280 nM T58921 C2JNM9 11234452 EC50 = 390 nM T58921 CBSO15 11234869 EC50 = 232 nM T58921 C7ROX3 11235560 IC50 = 483.06 nM T58921 CK4F7Q 11235859 IC50 = 520 nM T58921 CQ3C1F 11235892 EC50 > 3000 nM T58921 C2IBK8 11236542 IC50 > 15000 nM T58921 CBU98W 11236923 EC50 > 10000 nM T58921 CF31OJ 11237218 EC50 = 110 nM T58921 CGAI13 11237761 IC50 > 15000 nM T58921 C3B5FX 11243082 EC50 = 12302.69 nM T58921 CYO34T 11245626 EC50 > 5000 nM T58921 C8TP7X 11246061 EC50 ~ 5000 nM T58921 CG8IQ1 11246863 EC50 > 1000 nM T58921 CI07UN 11246958 EC50 ~ 5000 nM T58921 CL29MP 11247579 EC50 = 13 nM T58921 CP1X0G 11247654 IC50 = 88 nM T58921 C7C9MZ 11247664 EC50 > 3000 nM T58921 CBS49N 11247908 EC50 = 270 nM T58921 CY10BP 11247998 IC50 = 87 nM T58921 CVYS48 11248366 EC50 > 5000 nM T58921 C0PX1U 11248386 EC50 = 1000 nM T58921 C5VB4A 11248512 EC50 > 3000 nM T58921 CB68XN 11249025 EC50 = 6 nM T58921 C79VCR 11249385 IC50 = 1200 nM T58921 C73ZUY 11258935 EC50 = 570 nM T58921 C7LK0I 11258987 IC50 = 759 nM T58921 CRZ1Q9 11259404 EC50 = 179 nM T58921 CJ6ON0 11259787 EC50 = 28 nM T58921 CH9X1P 11260214 EC50 > 10000 nM T58921 CIA1W7 11262838 Ki = 251.19 nM T58921 C9J3DR 11271060 IC50 = 491 nM T58921 C7ZC0P 11271211 EC50 = 50 nM T58921 CYD12Z 11271514 EC50 = 30 nM T58921 CWH02S 11280270 EC50 > 1000 nM T58921 CK87RJ 11281114 EC50 = 360 nM T58921 CSOE29 11281767 EC50 = 200 nM T58921 CH69MT 11281802 EC50 > 3000 nM T58921 C19KDH 11282033 EC50 = 300 nM T58921 CNG61K 11282914 IC50 > 50000 nM T58921 C2O3WX 11283113 EC50 = 310 nM T58921 CP0H1J 11293283 EC50 > 1000 nM T58921 CDK79P 11293459 EC50 > 3000 nM T58921 C6T9OR 11294565 IC50 = 629 nM T58921 C5S6YO 11294660 IC50 = 1948 nM T58921 C4WDK1 11295072 EC50 = 5900 nM T58921 CFTW52 11295349 IC50 = 11.99 nM T58921 CMC6I8 11305717 EC50 = 9 nM T58921 CC81HS 11306364 IC50 = 1288.25 nM T58921 CDKC74 11306495 EC50 > 3000 nM T58921 C2KZ3M 11306745 EC50 = 478 nM T58921 CB12CE 11316788 EC50 = 228 nM T58921 CS60GO 11316811 EC50 = 295 nM T58921 C7Z1NC 11317347 EC50 > 3000 nM T58921 CUW3Q0 11317867 IC50 = 11 nM T58921 C0D7HU 11317892 IC50 = 440 nM T58921 CFQV09 11323235 EC50 = 25700 nM T58921 CUSY83 11327370 IC50 = 1790 nM T58921 C1OEB0 11328910 IC50 = 126 nM T58921 C9SB2M 11329011 IC50 = 1986 nM T58921 CIAP50 11329280 IC50 = 417 nM T58921 CSF2L4 11329304 EC50 = 60 nM T58921 CUL9I0 11335874 EC50 = 891.25 nM T58921 C6O3ZU 11339029 EC50 = 13 nM T58921 C2AK7F 11339346 EC50 = 1000 nM T58921 CMCD29 11339649 IC50 > 50000 nM T58921 C6WI0Z 11339975 IC50 = 6100 nM T58921 CP5F8D 11339979 IC50 = 51 nM T58921 C9B0LH 11340275 EC50 > 1000 nM T58921 CG91XM 11340322 EC50 > 3000 nM T58921 C0ABC9 11340513 EC50 = 6 nM T58921 CLFX14 11340991 IC50 = 2241 nM T58921 CI2J5W 11341085 IC50 = 1050 nM T58921 C0LU6S 11349723 EC50 > 1000 nM T58921 CATM03 11350008 IC50 > 50000 nM T58921 CQ7OF6 11351221 EC50 > 1000 nM T58921 CDL72P 11351238 EC50 = 1 nM T58921 C3CIB5 11351245 EC50 = 718 nM T58921 CEZG39 11351266 EC50 > 1000 nM T58921 C72GEN 11351550 EC50 > 3000 nM T58921 CL7D8V 11351980 EC50 > 3000 nM T58921 C9PAJ6 11352187 EC50 > 3000 nM T58921 CQN0X9 11352573 IC50 = 8.995 nM T58921 CET87Y 11352791 EC50 = 80 nM T58921 C8QTH7 11356973 EC50 = 12500 nM T58921 CKQ23T 11361486 EC50 = 243 nM T58921 C8VT0Y 11362757 IC50 = 1700 nM T58921 CZ30DH 11363106 EC50 = 7.7 nM T58921 CM7TX9 11363175 EC50 > 3000 nM T58921 C1UCN2 11363348 EC50 = 1000 nM T58921 CTA62X 11372106 EC50 ~ 5000 nM T58921 C4X1CW 11373702 EC50 > 5000 nM T58921 C5I4NE 11373767 EC50 = 152 nM T58921 CXHU81 11374318 EC50 = 1000 nM T58921 COZ01K 11374429 EC50 ~ 5000 nM T58921 C1JIT7 11374443 EC50 ~ 5000 nM T58921 C81BYX 11374677 EC50 = 9 nM T58921 CKE9R8 11374679 EC50 = 6 nM T58921 CDQ2M5 11374680 EC50 = 30 nM T58921 CJI2C6 11376123 EC50 = 1700 nM T58921 CZ5UX9 11381586 EC50 = 5400 nM T58921 C93MQC 11383635 IC50 > 15000 nM T58921 C5F8EY 11383668 EC50 = 48 nM T58921 C8V3HB 11384748 EC50 = 79 nM T58921 C5TZY0 11385663 IC50 = 3220 nM T58921 C3Z1LN 11386159 EC50 > 3000 nM T58921 C8WVM5 11386220 EC50 > 3000 nM T58921 C5OB8J 11386857 EC50 = 4220 nM T58921 C8X5PW 11393977 EC50 = 1130 nM T58921 C6SYD8 11396352 EC50 > 1000 nM T58921 CHRY56 11396567 EC50 = 644 nM T58921 CTU8G6 11397018 EC50 > 10000 nM T58921 C0TX7O 11397203 EC50 > 3000 nM T58921 CXIN63 11397705 EC50 > 10000 nM T58921 CGY28A 11405204 EC50 > 1000 nM T58921 CZB52S 11408244 IC50 = 2960 nM T58921 C34QBC 11408475 EC50 = 380.19 nM T58921 CX7W4S 11408502 EC50 > 3000 nM T58921 CPB8F6 11409173 EC50 = 111 nM T58921 CVG1X9 11414728 EC50 = 10500 nM T58921 C45UNR 11416269 IC50 > 10000 nM T58921 CKGU54 11418373 IC50 > 50000 nM T58921 CCV19Q 11418816 EC50 ~ 5000 nM T58921 CKA1D3 11418888 EC50 > 5000 nM T58921 CY0HO8 11418889 EC50 > 5000 nM T58921 CCAJ14 11418941 EC50 > 1000 nM T58921 C4KS1I 11419306 EC50 ~ 5000 nM T58921 CH5K6G 11419333 EC50 = 149 nM T58921 C6Q8FR 11419459 EC50 = 1200 nM T58921 CXJ72D 11419635 IC50 = 160 nM T58921 C2USN6 11419919 IC50 = 120 nM T58921 CI6ZE4 11419960 IC50 = 260 nM T58921 CMT65A 11421645 EC50 > 1000 nM T58921 CCD7X1 11421714 EC50 = 3 nM T58921 CXY7C1 11430619 EC50 > 5000 nM T58921 CZ3VT9 11430761 IC50 = 5600 nM T58921 C60KVM 11431103 EC50 = 4 nM T58921 C20VUO 11431152 IC50 = 1495 nM T58921 C5SKD2 11431192 EC50 = 121 nM T58921 CPGX09 11431289 EC50 = 407 nM T58921 C1OZ5D 11431625 EC50 = 465 nM T58921 CFU62G 11432162 EC50 = 303 nM T58921 C8XQL7 11438721 EC50 = 1600 nM T58921 C6FP3T 11441763 EC50 > 1000 nM T58921 CT4NR0 11442228 EC50 > 1000 nM T58921 C2ZVF9 11442294 EC50 = 8 nM T58921 CV5M3A 11442379 EC50 > 3000 nM T58921 CKF91A 11448976 IC50 > 50000 nM T58921 CO5M3W 11449787 IC50 > 50000 nM T58921 C8Q3LK 11452684 EC50 = 1000 nM T58921 C6ENV7 11453165 EC50 = 380 nM T58921 CE59YF 11453821 EC50 = 3 nM T58921 CFX90G 11454050 EC50 = 400 nM T58921 C6Q7UX 11454132 IC50 = 7900 nM T58921 C04YQX 11454155 EC50 = 2.1 nM T58921 CR5LM7 11463604 EC50 = 335 nM T58921 CJ7RT2 11463615 IC50 = 2700 nM T58921 C7XLZ9 11463785 EC50 = 5 nM T58921 C2Q6YV 11463996 IC50 > 50000 nM T58921 CF63PO 11464352 Ki = 81 nM T58921 CGIP81 11464448 EC50 = 234 nM T58921 C5PNY3 11464462 EC50 > 5000 nM T58921 C8X7SQ 11464817 EC50 = 1000 nM T58921 C4ZE1C 11465146 EC50 > 3000 nM T58921 CQT9S6 11466042 IC50 = 110 nM T58921 CW7U6D 11471872 EC50 = 1500 nM T58921 C6G7FO 11475460 EC50 > 1000 nM T58921 CN64KX 11475461 EC50 > 1000 nM T58921 C0V4HX 11476137 EC50 = 2 nM T58921 C7ZO8B 11476297 EC50 > 1000 nM T58921 CLZ5I1 11476382 IC50 > 15000 nM T58921 CI8FO6 11476916 EC50 > 3000 nM T58921 CSX3Z0 11477433 EC50 = 190 nM T58921 C7V4OW 11477633 EC50 > 5000 nM T58921 C83GWX 11477735 EC50 > 3000 nM T58921 CF3G8Y 11485037 EC50 > 5000 nM T58921 CQ6L9S 11486733 EC50 > 1000 nM T58921 C4S6JR 11488006 EC50 > 1000 nM T58921 CZ84QA 11488726 IC50 = 35 nM T58921 C6HO8J 11490050 EC50 > 1000 nM T58921 CQ9P3C 11497430 EC50 = 7.85 nM T58921 CL2V9K 11497604 EC50 > 10000 nM T58921 CF1AI0 11503439 EC50 > 10000 nM T58921 CU27FT 11503588 EC50 = 690 nM T58921 CK8NI4 11504194 EC50 = 950 nM T58921 CF36HJ 11508312 Ki = 515 nM T58921 C0JEO8 11511317 IC50 = 2707 nM T58921 CVMG07 11511500 EC50 = 3030 nM T58921 C39FAG 11511914 IC50 = 1368 nM T58921 CL4N9S 11512673 EC50 > 100000 nM T58921 CI8UO3 11520220 Ki = 912.01 nM T58921 C6MH7B 11524635 EC50 = 140 nM T58921 C0G5PF 11524965 EC50 = 200 nM T58921 CSX8A0 11525219 EC50 = 200 nM T58921 C68RSH 11525752 IC50 = 1199.5 nM T58921 CCJ50E 11526339 EC50 = 10560 nM T58921 CH14EK 11526493 EC50 = 2300 nM T58921 CDGL46 11530143 EC50 = 300 nM T58921 CRBI92 11532493 EC50 = 25 nM T58921 CU5A2J 11532616 EC50 > 10000 nM T58921 CT9Z0X 11539510 EC50 > 9700 nM T58921 C7BX1M 11540431 IC50 = 584 nM T58921 CC4T7S 11546596 EC50 = 15 nM T58921 C52AIP 11546956 IC50 = 12 nM T58921 CFCZ81 11553704 EC50 = 30 nM T58921 C70JZQ 11555240 EC50 = 2.3 nM T58921 CF5Q8T 11561245 EC50 = 550 nM T58921 C5H7FP 11563028 IC50 = 93 nM T58921 CSV9K4 11568541 EC50 = 20 nM T58921 C2IYQ4 11568811 EC50 = 18490 nM T58921 CKN39D 11569310 EC50 = 250 nM T58921 C9SJL1 11570226 EC50 = 45230 nM T58921 CRQ0W7 11575609 EC50 = 50 nM T58921 CE41FN 11577207 IC50 = 1452 nM T58921 CF2V1D 11583815 IC50 = 1580 nM T58921 C3GI8R 11585006 EC50 > 10000 nM T58921 CD6W0Y 11588094 Ki > 10000 nM T58921 CAKP71 11588179 EC50 > 10000 nM T58921 C1HG4A 11591164 EC50 = 10 nM T58921 CC15AQ 11592357 EC50 = 17 nM T58921 C0KY6R 11597691 EC50 = 660 nM T58921 CDR1Z3 11599646 EC50 = 32 nM T58921 C2ZP9O 11612623 IC50 = 1047 nM T58921 CE87MQ 11619439 EC50 = 6600 nM T58921 C5LVA3 11620018 IC50 = 127 nM T58921 C4M5SU 11620299 EC50 > 1000 nM T58921 CWOD63 11620575 EC50 = 2 nM T58921 CZ7FB6 11621704 Ki = 190.55 nM T58921 CCR92U 11624482 EC50 > 10000 nM T58921 CR30AV 11627288 IC50 = 129.12 nM T58921 C8CM4F 11627300 EC50 = 2190 nM T58921 C4ZR8D 11627859 EC50 = 630 nM T58921 C1GD3M 11628577 EC50 = 2810 nM T58921 CIT36S 11632586 EC50 = 80 nM T58921 C2JP8M 11633700 EC50 = 12300 nM T58921 C6JD1P 11635549 Ki = 138.04 nM T58921 C1FI8K 11635845 EC50 = 2160 nM T58921 CM6R1L 11640895 IC50 = 2072 nM T58921 CT7KW2 11647600 EC50 = 200 nM T58921 C6QZ4F 11649387 EC50 = 1140 nM T58921 C16CWN 11649783 EC50 > 10000 nM T58921 CY2DE9 11656305 IC50 = 2405 nM T58921 CDJ4F7 11656332 IC50 = 1282 nM T58921 C9H2TQ 11660029 EC50 = 28 nM T58921 CD0NU7 11663038 EC50 = 2820 nM T58921 CL7C1Z 11663931 EC50 > 10000 nM T58921 CQ2M8V 11669781 IC50 = 1900 nM T58921 CJNB58 11669835 EC50 = 70 nM T58921 CR9O3A 11670288 EC50 = 840 nM T58921 C1OH3U 11674387 EC50 = 549 nM T58921 C27FGM 11677450 EC50 = 290 nM T58921 CHA36Y 11678044 IC50 = 2024 nM T58921 C6H8PJ 11678481 EC50 = 70000 nM T58921 C91EWR 11678534 EC50 = 2 nM T58921 C2CHW3 11682417 Ki = 695 nM T58921 C8MU1C 11683336 EC50 = 4900 nM T58921 CQ43HN 11685800 Ki = 54.95 nM T58921 CX0TY6 11688434 EC50 = 700 nM T58921 C0NI8S 11690159 EC50 = 90 nM T58921 CR5X7O 11697915 EC50 = 50 nM T58921 CDN9H0 11698089 EC50 = 30 nM T58921 CS3PO8 11698476 EC50 > 4900 nM T58921 CD43TA 11698802 EC50 = 102 nM T58921 C3FIK4 11704026 EC50 = 200 nM T58921 C90QUD 11704765 EC50 = 80 nM T58921 CR46YH 11705832 IC50 = 2409 nM T58921 CZ1VX2 11710179 EC50 > 10000 nM T58921 C2WQ1O 11711595 EC50 = 1900 nM T58921 CW1VA6 11712195 EC50 = 300 nM T58921 C5AX8M 11712774 IC50 = 3968 nM T58921 C2UY7P 11712873 IC50 = 105 nM T58921 CVZY96 11721801 Ki = 100 nM T58921 CRY41K 11723307 EC50 > 100000 nM T58921 C5UIL7 11729738 EC50 = 6200 nM T58921 C6C9HF 11741962 IC50 = 1500 nM T58921 C5FYH0 11742116 EC50 = 130 nM T58921 CLR1Y7 11750299 EC50 = 274 nM T58921 CNQ6O1 11750720 EC50 > 1000 nM T58921 C51EZG 11750812 IC50 = 220 nM T58921 CR7Y2E 11751021 IC50 = 345.94 nM T58921 C2FNH3 11751223 EC50 = 1000 nM T58921 CHB64T 11751299 EC50 = 359 nM T58921 C7V0DE 11751301 EC50 = 0.55 nM T58921 C0Q4XH 11753952 Ki = 3.1 nM T58921 C35DKP 11754345 EC50 = 30902954.33 nM T58921 CLE5P8 11754583 IC50 > 15000 nM T58921 C7O6FH 11755396 EC50 = 6456542.29 nM T58921 C18XBA 11755655 EC50 > 3000 nM T58921 CL4EK8 11755968 EC50 = 56234132.52 nM T58921 C58DMZ 11757696 EC50 = 40 nM T58921 CKWA01 11772573 IC50 > 50000 nM T58921 CPV6E2 11774184 EC50 = 41 nM T58921 C9D4OH 11774537 EC50 = 4 nM T58921 C7WQ9E 11774595 EC50 = 180 nM T58921 CBV25C 11774828 EC50 = 836 nM T58921 C95FTM 11774965 EC50 = 2900 nM T58921 CE27GQ 11775099 EC50 = 390 nM T58921 C3EXH7 11775225 EC50 = 2160 nM T58921 CA0LW8 11784454 EC50 = 10.96 nM T58921 CX5YP8 11784860 EC50 = 15 nM T58921 CW8R9F 11785036 EC50 = 640 nM T58921 CZ0B4P 11785404 IC50 = 1784 nM T58921 CT54GI 11799712 Ki = 144.54 nM T58921 C8BQN9 11800577 Ki = 120.23 nM T58921 C9YT0O 11800617 EC50 = 1.445 nM T58921 CHUA47 11801489 Ki = 12.3 nM T58921 C7J1QY 11802274 Ki = 53.7 nM T58921 C5N4VH 11811337 EC50 = 3000 nM T58921 C5MJ8U 11811825 EC50 = 460 nM T58921 CZ52VY 11813713 Ki = 4.6 nM T58921 CL7V4Z 11826628 EC50 = 280 nM T58921 C63HSV 11845112 EC50 > 10000 nM T58921 CD2EH5 11845115 EC50 > 10000 nM T58921 CWG17X 11845116 EC50 = 1000 nM T58921 CX6WA3 11845117 EC50 = 2500 nM T58921 C6YBA3 11845277 EC50 = 300 nM T58921 C7F0IH 11845280 EC50 = 220 nM T58921 C1TM2W 11845281 EC50 = 210 nM T58921 C5L1RK 11845282 EC50 = 50 nM T58921 CAO2Q1 11948655 EC50 = 480 nM T58921 C38KZG 11978565 EC50 = 13000 nM T58921 CEW4G1 11978566 EC50 = 12000 nM T58921 CQH67B 11978567 EC50 = 5500 nM T58921 CJO9Z6 11978569 EC50 = 6200 nM T58921 C1AOP8 11978570 EC50 = 13000 nM T58921 C1CBW0 11992126 EC50 = 642 nM T58921 COPI61 11997929 EC50 > 10000 nM T58921 CB45PX 12082255 EC50 = 7600 nM T58921 C9AG1K 12082256 EC50 = 4800 nM T58921 CVL12Z 12109364 EC50 = 200 nM T58921 CQ36YX 12109366 IC50 = 400 nM T58921 CQ6R7S 12111897 Ki = 1500 nM T58921 CVIZ19 12112546 IC50 = 110 nM T58921 CV2OW5 12132847 EC50 > 10000 nM T58921 CWL9C6 12967684 EC50 = 2800 nM T58921 CA19MJ 13965473 EC50 = 3100 nM T58921 CQSK24 14163455 IC50 = 110 nM T58921 CS82RI 14427412 EC50 = 3600 nM T58921 CH62MC 14626814 EC50 = 230 nM T58921 CKMB21 14626863 EC50 = 2490 nM T58921 CFK4L0 14730796 IC50 = 124000 nM T58921 CD7R9F 15069292 EC50 = 400 nM T58921 C7GE4V 15069295 EC50 = 1900 nM T58921 CDM80R 15069396 EC50 = 260 nM T58921 C0LH2E 15942850 EC50 = 300 nM T58921 C6J5WN 15951505 IC50 = 18 nM T58921 C5KP7J 15979459 EC50 = 5000 nM T58921 CF6I7X 15981441 EC50 = 71 nM T58921 CDFT16 15984029 EC50 = 30 nM T58921 CEL3S6 16007090 EC50 = 1582 nM T58921 CVX7D4 16036020 EC50 = 2.6 nM T58921 C9T1QR 16036021 EC50 = 15 nM T58921 C19HBE 16036133 EC50 = 4.5 nM T58921 CT3VA7 16036134 EC50 = 7.5 nM T58921 CET7R0 16036257 EC50 = 1.1 nM T58921 CWE62Y 16038358 EC50 = 28 nM T58921 C8J0TE 16040328 EC50 = 140 nM T58921 CO5B2T 16043249 EC50 > 10000 nM T58921 CY13OS 16046718 EC50 = 8000 nM T58921 CPY13K 16046721 EC50 = 2000 nM T58921 CTP15X 16046722 EC50 = 4000 nM T58921 C7AIM9 16048150 EC50 = 11 nM T58921 CE1A9C 16058409 EC50 > 10000 nM T58921 C05RLT 16058623 EC50 = 47.7 nM T58921 C4ENU6 16058624 EC50 = 208 nM T58921 C8H7NA 16064438 EC50 = 12 nM T58921 C25QGK 16066144 EC50 = 180 nM T58921 C5V0ZY 16085979 EC50 = 674 nM T58921 CD3K9X 16085980 IC50 = 5.998 nM T58921 CY1Q3Z 16085981 EC50 = 5 nM T58921 C1F6CM 16085982 EC50 = 355 nM T58921 C97HJA 16085983 EC50 = 112 nM T58921 CE3HN1 16085984 EC50 = 46 nM T58921 C2F4AJ 16085985 IC50 = 15 nM T58921 CE4Q7N 16085986 EC50 = 4 nM T58921 CXYF29 16085987 EC50 = 402 nM T58921 CPQ2K9 16085988 IC50 = 19 nM T58921 CF4J1K 16090330 EC50 = 320 nM T58921 CU63PB 16090857 EC50 = 2210 nM T58921 CA51QP 16090858 EC50 = 210 nM T58921 C8O1HI 16090859 EC50 = 470 nM T58921 CMKI28 16090878 EC50 = 3470 nM T58921 CJC53L 16090879 EC50 = 650 nM T58921 CJ3D4H 16109183 EC50 = 1870 nM T58921 CJ38DY 16109187 EC50 > 10000 nM T58921 CS8NF6 16109190 EC50 > 10000 nM T58921 C9IO5Z 16109193 EC50 > 25000 nM T58921 CU0BK1 16109199 EC50 > 10000 nM T58921 C2S0TO 16109209 EC50 > 25000 nM T58921 C7V9EL 16109210 EC50 > 10000 nM T58921 CP0SB8 16110418 EC50 > 10000 nM T58921 C4W5IY 16110419 EC50 = 181970.09 nM T58921 CHJ4Z3 16110420 EC50 = 338844.16 nM T58921 C2TO3Q 16110421 EC50 = 1071519.31 nM T58921 CDVL80 16110424 EC50 = 467735.14 nM T58921 C3X2WM 16110425 EC50 = 1778279.41 nM T58921 C4T0RO 16110426 EC50 = 602559.59 nM T58921 CT78IG 16110427 EC50 = 1445439.77 nM T58921 CYZ74P 16110428 EC50 = 1819700.86 nM T58921 C7IL6H 16110429 EC50 = 117489.76 nM T58921 CE91XP 16110436 EC50 = 1548816.62 nM T58921 C9W4KS 16110437 EC50 = 245470.89 nM T58921 C2OZJ4 16110438 EC50 = 1380384.26 nM T58921 C6FA1K 16110439 EC50 = 1819700.86 nM T58921 CI05UK 16110440 EC50 = 2089296.13 nM T58921 CI4Z8S 16110441 EC50 = 1047128.55 nM T58921 C2UJ6Y 16110442 EC50 = 3388441.56 nM T58921 CBW78Z 16110443 EC50 = 1819700.86 nM T58921 CE19FD 16110444 EC50 = 562341.33 nM T58921 C7F0IX 16110482 EC50 = 20892961.31 nM T58921 C3PXV5 16110483 EC50 = 2691534.8 nM T58921 C5WZ4Y 16110484 EC50 = 1047128.55 nM T58921 CCM5G9 16110485 EC50 = 1148153.62 nM T58921 C0N6VP 16110486 EC50 = 22387211.39 nM T58921 C5NX0T 16110487 EC50 = 3090295.43 nM T58921 CC24LB 16110489 EC50 = 3467368.5 nM T58921 CNU63E 16110490 EC50 = 23988329.19 nM T58921 CQ0T9X 16110492 EC50 = 1148153.62 nM T58921 CF15DS 16110493 EC50 = 1348962.88 nM T58921 CTC3I5 16110494 EC50 = 22387211.39 nM T58921 CNS35L 16110511 EC50 = 162181.01 nM T58921 CXQD14 16110512 EC50 = 1000000 nM T58921 C4TO1G 16110514 EC50 = 125892.54 nM T58921 CZ5RS7 16110516 EC50 = 660693.45 nM T58921 CU1S0A 16110517 EC50 = 616595 nM T58921 CO5D1F 16110518 EC50 = 812830.52 nM T58921 CB8Q6G 16110519 EC50 = 181970.09 nM T58921 CW4V2X 16110524 EC50 = 5623413.25 nM T58921 CT35DL 16110525 EC50 = 2089296.13 nM T58921 C4F5EU 16110532 EC50 = 1000000 nM T58921 CZ3AN2 16110534 EC50 = 14791083.88 nM T58921 CXN40P 16110535 EC50 = 5623413.25 nM T58921 C0KL4A 16220189 Ki = 3.42 nM T58921 CE71MI 16220190 EC50 = 1100 nM T58921 CR3C1Q 16222636 EC50 = 4000 nM T58921 C49IER 16722365 EC50 = 980 nM T58921 CD7L4Z 16726113 EC50 > 1000 nM T58921 C92NRU 16727109 EC50 > 1610 nM T58921 CM9YZ5 16739272 IC50 = 240 nM T58921 CN6CU3 16739344 EC50 = 1030 nM T58921 CD65RZ 16742591 EC50 > 1000 nM T58921 C8LPX0 16747684 EC50 = 800 nM T58921 CCPS15 16753427 IC50 = 3500 nM T58921 C83AOY 17894227 Ki = 32 nM T58921 CFS4T7 17894542 EC50 = 70 nM T58921 CXS40D 17950432 EC50 = 458 nM T58921 CW4K9X 17984540 IC50 = 91 nM T58921 CQ2N0I 18003428 IC50 = 30 nM T58921 CW29KQ 18003431 EC50 = 16 nM T58921 CHB98X 18003446 EC50 = 123 nM T58921 C8WQ6D 18003447 EC50 = 18 nM T58921 CAOS67 18003481 IC50 = 2 nM T58921 CA32RT 18003618 IC50 = 3 nM T58921 CAO59H 18438761 EC50 = 12 nM T58921 CJNB84 18442897 EC50 = 2050 nM T58921 CLE7Y9 18442898 EC50 = 2110 nM T58921 CT1CI8 18442899 EC50 = 3020 nM T58921 CY0L2U 18442903 EC50 = 1120 nM T58921 CX18MV 18442904 EC50 = 90 nM T58921 CAS20N 18442912 EC50 = 150 nM T58921 C9WU4K 18442916 EC50 = 830 nM T58921 C6BKW9 18442917 EC50 = 3430 nM T58921 CL94NS 18654313 EC50 = 2620 nM T58921 CF9BK7 18701962 Ki = 34 nM T58921 CP8GD2 18702001 Ki = 32 nM T58921 C2GN1I 18766436 EC50 = 110 nM T58921 CBLA15 18794804 Ki = 15 nM T58921 CO4QB0 18944089 Ki = 0.4 nM T58921 CA82PW 19008901 EC50 = 574 nM T58921 CT7ED5 19008935 EC50 = 2200 nM T58921 CYK70R 19080384 Ki = 1100 nM T58921 CL3AP9 19792109 EC50 = 5010 nM T58921 CR5T0X 20356227 EC50 > 10000 nM T58921 C2C8VM 20765803 EC50 = 200 nM T58921 C3G8NO 20765805 EC50 = 400 nM T58921 CXGK50 20765807 EC50 = 1000 nM T58921 CW3G2Y 20777233 EC50 = 4400 nM T58921 C1LOC3 21054974 EC50 = 1100 nM T58921 CV7UB3 21054981 EC50 = 1500 nM T58921 COLV42 21054982 EC50 = 1800 nM T58921 CP3RI0 21054984 EC50 = 100 nM T58921 CNW9C5 21054988 EC50 = 2100 nM T58921 C5BM3O 21055003 EC50 = 5000 nM T58921 CX2FC0 21101227 EC50 = 1200 nM T58921 CT96QD 21357774 EC50 = 10 nM T58921 C7ONA8 21700391 Ki = 15.49 nM T58921 C51VRK 21700407 Ki = 0.9333 nM T58921 CLY6W8 21700419 EC50 = 0.912 nM T58921 CAH60U 21700457 EC50 = 1.413 nM T58921 CGY69K 21700480 EC50 = 416.87 nM T58921 CU8S1L 21700481 Ki = 3.236 nM T58921 CF0M9Q 21700497 Ki = 3.388 nM T58921 CX48VU 21866618 EC50 = 3000 nM T58921 CES61V 21866640 EC50 = 10000 nM T58921 CY0TR2 21866670 EC50 = 10000 nM T58921 CX2J7L 21866721 EC50 = 10000 nM T58921 C3SWL4 21866734 EC50 = 1000 nM T58921 CEMT42 21866801 EC50 = 3000 nM T58921 CMGS41 21866827 EC50 = 300 nM T58921 CX05LN 21866931 EC50 = 300 nM T58921 CGHF16 21866936 EC50 = 3000 nM T58921 CU0IJ4 21928218 EC50 > 10000 nM T58921 C2O4BZ 21928229 EC50 = 910 nM T58921 CEWR84 21942712 EC50 = 68 nM T58921 C48BOL 21942716 EC50 = 347 nM T58921 CU58VO 21942721 EC50 = 3180 nM T58921 COKU53 21942723 EC50 = 104 nM T58921 CZF52L 21942731 EC50 = 1860 nM T58921 CC98SZ 21942737 EC50 = 306 nM T58921 C4T1SY 21942738 EC50 = 45 nM T58921 CAC2U8 21942751 EC50 > 10000 nM T58921 CY58SO 21942772 EC50 = 617 nM T58921 CFBM32 21942781 EC50 = 12 nM T58921 CS2U1Y 21942782 EC50 = 52 nM T58921 CFRH71 21985914 Ki = 1090 nM T58921 CI40KU 22087541 EC50 = 36 nM T58921 CN97KU 22087544 EC50 = 359 nM T58921 C6SQ5I 22087586 EC50 = 52 nM T58921 C17ZPC 22087654 EC50 = 705 nM T58921 CB2G3Y 22087658 EC50 = 267 nM T58921 CNBL28 22148735 IC50 = 19 nM T58921 CV0MX1 22229246 EC50 = 815 nM T58921 CU6YG1 22229249 EC50 > 3000 nM T58921 C28MRJ 22229258 EC50 > 3000 nM T58921 C4L5TH 22229292 EC50 > 3000 nM T58921 CSAX56 22229323 EC50 > 3000 nM T58921 C8MT5I 22261152 EC50 = 800 nM T58921 CM93FV 22279993 IC50 = 7570 nM T58921 CGVR07 22280001 IC50 > 10000 nM T58921 CE3OI9 22280016 IC50 = 21600 nM T58921 C1BG7A 22280047 IC50 < 11100 nM T58921 C1G2OH 22280062 IC50 = 13800 nM T58921 C14YDT 22280073 IC50 = 9120 nM T58921 CDQ0Y6 22280103 IC50 = 5559.04 nM T58921 C0VET7 22280114 IC50 = 33265.96 nM T58921 C7IW1Y 22280124 IC50 < 11100 nM T58921 COA0S5 22280155 IC50 > 11000 nM T58921 CVH3O8 22280178 IC50 > 10000 nM T58921 CK1ZY7 22504766 IC50 > 10000 nM T58921 C2P7OG 22504815 IC50 > 10000 nM T58921 CDK75I 22504857 IC50 > 10000 nM T58921 CO0UC5 22504899 IC50 > 10000 nM T58921 CHD4Z0 22504917 IC50 = 8660 nM T58921 CU4JP1 22610192 EC50 = 43 nM T58921 CSZ7H9 22610195 EC50 = 37 nM T58921 CE5Z8K 22610208 EC50 = 113 nM T58921 CS0HE9 22727983 EC50 = 7900 nM T58921 CE06NF 22728012 EC50 = 3300 nM T58921 CG9O8Q 22928715 EC50 = 1900 nM T58921 CD9QL8 22993865 EC50 = 600 nM T58921 CXJ7I3 22993874 IC50 = 2000 nM T58921 C3K4ZA 22993886 IC50 = 66 nM T58921 CG23ZP 23111663 EC50 = 10000 nM T58921 CT38PB 23111732 EC50 = 5260 nM T58921 CJ5NM3 23249734 EC50 = 300 nM T58921 C8M3RA 23362219 Ki = 6000 nM T58921 CM1TL6 23362228 Ki = 600 nM T58921 CNV6R2 23362229 Ki = 33 nM T58921 CAW5I4 23362235 Ki = 37 nM T58921 CNXB90 23402689 EC50 = 2370 nM T58921 C8Z5MA 23402692 EC50 = 4 nM T58921 CU18VJ 23402759 IC50 = 70 nM T58921 CSLH35 23402760 IC50 = 160 nM T58921 CBZ85M 23402773 EC50 = 4200 nM T58921 C1PBI5 23402831 EC50 = 7330 nM T58921 C14KIP 23402832 IC50 = 712 nM T58921 C7HSI3 23515186 EC50 = 1000 nM T58921 C2MX7P 23529368 EC50 = 4 nM T58921 C10TAO 23553234 EC50 = 580 nM T58921 C7NRY5 23572034 Ki = 1500 nM T58921 CEJ1S4 23628240 EC50 = 160 nM T58921 CL6AD8 23628247 IC50 > 10000 nM T58921 CS26KY 23648476 EC50 = 506 nM T58921 CO6EC1 23648933 EC50 = 220 nM T58921 CX8W7E 23649183 EC50 = 2819 nM T58921 C9NPQ4 23651402 EC50 = 271 nM T58921 CD7HN9 23651403 EC50 = 1740 nM T58921 C18CXM 23656548 EC50 > 10000 nM T58921 C0WDH8 23657636 EC50 = 6 nM T58921 C6CZ1W 23661590 EC50 = 1310 nM T58921 CT43OQ 23661729 EC50 = 5500 nM T58921 C0VKM5 23672434 Ki = 969 nM T58921 CZPJ84 23674509 Ki = 1030 nM T58921 CAP8K7 23676879 Ki = 6690 nM T58921 CY82MF 23678396 EC50 = 340 nM T58921 C0D2NA 23683103 Ki > 10000 nM T58921 C7W8GM 23684387 Ki > 10000 nM T58921 C8WL4M 23684920 Ki = 4390 nM T58921 C9H4WT 23686961 EC50 = 3981.07 nM T58921 CF04QP 23690285 Ki > 10000 nM T58921 C5S7GF 23703312 EC50 = 617 nM T58921 CI5P0C 23874497 EC50 = 1200 nM T58921 CV6A3P 24210649 IC50 = 434 nM T58921 CR02NF 24739090 EC50 = 50 nM T58921 CTE1N2 24748569 EC50 > 10000 nM T58921 C56SGF 24754924 IC50 = 38.99 nM T58921 CNBV74 24759099 EC50 = 6 nM T58921 C73QEI 24808475 EC50 > 10000 nM T58921 CLV9T5 24816384 EC50 = 3000 nM T58921 C70QHI 24828802 EC50 = 30000 nM T58921 C15NSJ 24828803 EC50 = 52000 nM T58921 CO31MA 24828805 EC50 = 49000 nM T58921 CW51RK 24828806 EC50 = 38000 nM T58921 CVDQ19 24849963 EC50 = 3 nM T58921 C48SQZ 24875337 EC50 = 3443 nM T58921 C3E7IZ 24882613 EC50 = 70 nM T58921 CP1EM0 24890166 EC50 = 320 nM T58921 C34OKV 24890167 EC50 = 710 nM T58921 C0PYD9 24890168 EC50 > 10000 nM T58921 C5Q1GX 24890333 EC50 = 110 nM T58921 C5FV9O 24890334 EC50 = 140 nM T58921 C0P4RE 24890336 EC50 > 10000 nM T58921 CMU63N 24890509 EC50 = 190 nM T58921 CF57SZ 24890510 EC50 = 1100 nM T58921 C13XCE 24890511 EC50 = 120 nM T58921 CKT23B 24890512 EC50 = 280 nM T58921 C94RLU 24890513 EC50 = 2300 nM T58921 C7LTC8 24890684 EC50 = 620 nM T58921 C3MDU5 24890685 EC50 = 1300 nM T58921 CV1Q0H 24936142 EC50 = 84 nM T58921 C6ZG0A 24936147 EC50 = 40 nM T58921 CC13ZW 24936148 EC50 = 69 nM T58921 C8PD2Z 24941254 IC50 = 7943.28 nM T58921 C1P6WN 24949595 EC50 = 300 nM T58921 C17UHS 24949596 EC50 = 400 nM T58921 C1CG8I 24949919 EC50 = 1000 nM T58921 CX1WF4 24963031 EC50 = 140 nM T58921 CU41PY 25008799 Ki = 18 nM T58921 C21QHZ 25014794 EC50 = 102 nM T58921 CQWZ49 25032861 EC50 = 1100 nM T58921 C68JNV 25034259 EC50 > 10000 nM T58921 CD6L4X 25034260 EC50 = 1100 nM T58921 C0U2EC 25034324 EC50 = 1700 nM T58921 C93YUF 25034325 EC50 = 2400 nM T58921 C43JFV 25034326 EC50 = 2500 nM T58921 CEZG05 25034327 EC50 = 1100 nM T58921 CS8X2F 25034328 EC50 = 900 nM T58921 CG37TO 25034329 EC50 = 1300 nM T58921 C8GZR9 25034330 EC50 = 1900 nM T58921 CQ0AW7 25034407 EC50 = 200 nM T58921 C5DUK6 25034408 EC50 = 1200 nM T58921 C2FK3P 25034409 EC50 > 10000 nM T58921 CU2NI4 25034410 EC50 = 100 nM T58921 CYQ83S 25034411 EC50 = 100 nM T58921 CSP52M 25034412 EC50 = 1500 nM T58921 CC9TW1 25034413 EC50 = 100 nM T58921 CV7DO8 25034475 EC50 = 1500 nM T58921 C9M6CG 25034476 EC50 = 100 nM T58921 C54PWJ 25058068 EC50 = 2 nM T58921 CF98EG 25071332 EC50 = 38 nM T58921 CAOE29 25104183 EC50 = 639 nM T58921 C6WL7Z 25107241 EC50 = 300 nM T58921 C8CAY3 25110733 EC50 = 3060 nM T58921 CZ8AR6 25110744 EC50 = 1060 nM T58921 CB01VE 25113156 EC50 = 5930 nM T58921 CU78IR 25114869 EC50 = 121 nM T58921 CKEV40 25114870 EC50 = 1890 nM T58921 CI53RL 25114871 EC50 = 36 nM T58921 CU1T2F 25114873 EC50 = 40 nM T58921 CDA68R 25115099 EC50 = 2940 nM T58921 C4Q1WY 25115101 EC50 = 1610 nM T58921 C0BT6Z 25115103 EC50 = 175 nM T58921 CUW4D0 25115277 EC50 = 134 nM T58921 CZH49S 25115278 EC50 = 201 nM T58921 CWJ0T7 25115333 EC50 = 46 nM T58921 CG1TV7 25115504 EC50 = 68 nM T58921 CMK0A5 25115507 EC50 = 40 nM T58921 C6RT7Y 25115556 EC50 = 279 nM T58921 CR3FK4 25115789 EC50 = 25400 nM T58921 CF31BP 25115790 EC50 = 220 nM T58921 CDF4J5 25115793 EC50 = 1160 nM T58921 C2H5QL 25116020 EC50 = 816 nM T58921 CZW5M7 25116021 EC50 = 740 nM T58921 CT93BD 25116250 EC50 = 606 nM T58921 CRNB78 25116251 EC50 = 38600 nM T58921 C2M6GN 25116484 EC50 = 28100 nM T58921 CI9SL3 25116487 EC50 = 3190 nM T58921 C4M6ZY 25116726 EC50 = 2730 nM T58921 CWQ54L 25116728 EC50 = 41400 nM T58921 C5F3XY 25116813 EC50 = 139 nM T58921 C7Y4EV 25116953 EC50 = 6930 nM T58921 CHD2G4 25116956 EC50 = 1850 nM T58921 CXE3I5 25116957 EC50 = 25100 nM T58921 C57LQZ 25117176 EC50 = 26 nM T58921 C1J5LQ 25117396 EC50 = 10 nM T58921 C3NU1E 25132561 EC50 = 3290 nM T58921 CJ06KN 25132562 EC50 = 37400 nM T58921 C5DV8Z 25147673 EC50 = 15 nM T58921 CYFQ56 25147837 EC50 = 250 nM T58921 CX05GL 25147838 EC50 = 1 nM T58921 CJAC29 25147839 EC50 = 1 nM T58921 CASK45 25147840 EC50 = 170 nM T58921 C4OVN0 25147933 EC50 = 1 nM T58921 CXR1L0 25148011 EC50 = 1740 nM T58921 C9RSZ4 25148012 EC50 = 1 nM T58921 C7NXK8 25148013 EC50 = 1620 nM T58921 CIN0X4 25148014 EC50 = 1120 nM T58921 COS02A 25148015 EC50 = 100 nM T58921 CX25ZB 25148016 EC50 = 1 nM T58921 C1L6RT 25148090 EC50 = 160 nM T58921 C2I9DM 25149038 EC50 = 1260 nM T58921 CC9GO5 25149124 EC50 = 350 nM T58921 C8N3SX 25149125 EC50 = 1 nM T58921 C0Q7ZR 25149126 EC50 = 420 nM T58921 CM4F1V 25149127 EC50 = 960 nM T58921 C8JA1W 25149128 EC50 = 3550 nM T58921 CSMT48 25149129 EC50 = 1 nM T58921 CX97GA 25164959 EC50 = 1 nM T58921 CZ6PL9 25164960 EC50 = 1 nM T58921 C45WHD 25165162 EC50 = 2 nM T58921 CZF5B0 25165359 IC50 < 1 nM T58921 C7W3IH 25165560 EC50 = 9 nM T58921 CZ4TN9 25165638 IC50 = 25 nM T58921 CER49X 25165639 IC50 = 54 nM T58921 CBPX25 25166738 EC50 = 140 nM T58921 C3HAY5 25166740 EC50 = 4 nM T58921 C4WNU0 25166741 EC50 = 4 nM T58921 CPE1I4 25166743 EC50 = 94 nM T58921 CS03PW 25166956 IC50 = 3 nM T58921 CBRJ15 25167638 EC50 = 40 nM T58921 C72AEW 25167766 EC50 = 4 nM T58921 C0PAE1 25179516 EC50 = 3700 nM T58921 C5RBW3 25179712 IC50 = 1500 nM T58921 C54DIT 25179907 EC50 = 8300 nM T58921 CW86SI 25181477 IC50 = 44000 nM T58921 C71PGV 25206537 IC50 = 11700 nM T58921 C64FTI 25211572 EC50 = 3 nM T58921 CZ9H6S 25211874 EC50 = 2060 nM T58921 CT51NS 25211876 IC50 = 3162.28 nM T58921 CSWB02 25211877 IC50 = 3162.28 nM T58921 CRVP72 25227445 EC50 = 6620 nM T58921 C50YNC 25243830 EC50 = 41 nM T58921 CC71LU 25256813 IC50 = 1600 nM T58921 CUPT26 25261785 EC50 = 3500 nM T58921 CK09UM 25261937 EC50 = 4460 nM T58921 C6S8NL 25261938 EC50 = 4790 nM T58921 C73GBQ 25262090 EC50 = 6130 nM T58921 CMH0D6 25262091 EC50 >= 50000 nM T58921 C2H7ML 25262242 EC50 = 4940 nM T58921 CK5X2S 25262243 EC50 = 4470 nM T58921 CJAO04 25262244 EC50 >= 50000 nM T58921 C0G6BR 25262245 EC50 >= 50000 nM T58921 CR3E5T 25263358 IC50 > 10000 nM T58921 CU68GV 25263359 IC50 = 5011.87 nM T58921 COFY03 25263360 IC50 = 3981 nM T58921 CL6SG8 25263361 IC50 = 2511.89 nM T58921 CJW5Z8 25263362 IC50 = 6309.57 nM T58921 C2YU5K 25263363 IC50 = 3162.28 nM T58921 CB70OD 25263364 IC50 = 3981.07 nM T58921 CE7MW2 25263365 IC50 > 10000 nM T58921 CAM4D7 25263366 IC50 = 5011.87 nM T58921 C5KJS4 25263367 IC50 = 5011.87 nM T58921 CT5R1F 25263368 IC50 = 7943.28 nM T58921 CO16NL 25263369 IC50 = 7943.28 nM T58921 C6NSB5 25263370 IC50 = 6309.57 nM T58921 C7KPY3 25263371 IC50 = 3162.28 nM T58921 CLS1I8 25263372 IC50 = 3981.07 nM T58921 C7U4IG 25263373 IC50 = 5011.87 nM T58921 CJ7NW1 25263374 IC50 = 1995 nM T58921 CY09AD 25263375 IC50 = 1258.93 nM T58921 CPT2M7 25263376 IC50 = 1584.89 nM T58921 C3J6IA 25263377 IC50 = 2511.89 nM T58921 CJG62V 25263378 IC50 = 1584.89 nM T58921 CV5S1G 25263379 IC50 = 10000 nM T58921 C5QA6B 25263380 IC50 = 2511.89 nM T58921 CF49OS 25263381 IC50 = 1995.26 nM T58921 CZDA26 25263382 IC50 = 7943.28 nM T58921 CG59MP 25263383 IC50 = 1000 nM T58921 CD9EZ2 25263384 IC50 = 794.33 nM T58921 C10NLX 25263385 IC50 = 5011.87 nM T58921 C50GAO 25263386 IC50 = 1995.26 nM T58921 C8KCW3 25263387 IC50 = 3981.07 nM T58921 CJST96 25263388 IC50 = 2511.89 nM T58921 CW6U1B 25263389 EC50 > 1000 nM T58921 CKMR46 25263390 EC50 > 1000 nM T58921 CZ0CO2 25263391 EC50 > 10000 nM T58921 C3P9KJ 25263392 EC50 > 10000 nM T58921 CA8JG2 25263393 EC50 > 10000 nM T58921 C9B0PG 25263394 EC50 > 10000 nM T58921 CE35MH 25263395 EC50 > 10000 nM T58921 C3RG0W 25263396 EC50 > 10000 nM T58921 C19DVJ 25263397 EC50 > 10000 nM T58921 C3FGA6 25263398 EC50 > 10000 nM T58921 C04WDJ 25263399 EC50 > 10000 nM T58921 CHL2X3 25263400 EC50 > 10000 nM T58921 CGZL24 25263401 EC50 = 2.1 nM T58921 CUMZ05 25263402 EC50 = 1 nM T58921 CPO0U4 25263403 EC50 = 0.3 nM T58921 CFS9A2 25263404 EC50 = 0.19 nM T58921 CC29YB 25263405 EC50 = 0.36 nM T58921 CD9SV4 25263406 EC50 = 0.31 nM T58921 CJ6L2O 25263407 EC50 = 0.1 nM T58921 CBGE67 25263408 EC50 = 0.54 nM T58921 C08EKY 25263409 EC50 = 5 nM T58921 CH5PV6 25263410 EC50 = 6.8 nM T58921 C6F0WS 25263411 EC50 = 28 nM T58921 C78DHO 25263412 EC50 = 20 nM T58921 CBM0U5 25263413 EC50 = 5.2 nM T58921 CD5UF1 40484423 Ki = 169.1 nM T58921 C6Z2KG 42604838 EC50 = 110 nM T58921 CNU8Q0 42608446 Ki = 33 nM T58921 CR3ZD5 42613829 EC50 = 6360 nM T58921 CX70AK 42625720 EC50 = 3500 nM T58921 CW36AR 42625721 EC50 = 1070 nM T58921 CX6D9E 42625795 EC50 = 2120 nM T58921 C2TK3Z 42625796 EC50 = 370 nM T58921 CRLG64 42625797 EC50 = 120 nM T58921 C3UKN7 42625798 EC50 = 420 nM T58921 CNE6U4 42625799 EC50 = 540 nM T58921 CVAN68 42625871 EC50 = 100 nM T58921 CG8K1S 42625874 EC50 > 10000 nM T58921 C86XNA 42625875 EC50 = 2070 nM T58921 CW0A6E 42625952 EC50 = 430 nM T58921 C67UGQ 42625953 EC50 = 510 nM T58921 CC6YK7 42625954 EC50 = 2800 nM T58921 C83VLK 42625955 EC50 = 300 nM T58921 CC81PK 42625956 EC50 > 10000 nM T58921 C04ROU 42626028 EC50 = 470 nM T58921 CI4VG0 42626029 EC50 = 100 nM T58921 CIJ3H9 42626030 EC50 = 50 nM T58921 CAF31V 42641524 EC50 = 251.19 nM T58921 CL18EJ 44132007 EC50 = 158.49 nM T58921 CX7W2E 44132009 EC50 = 10 nM T58921 COZ56I 44132010 EC50 = 7.943 nM T58921 C6GBX4 44132012 EC50 = 5.012 nM T58921 CANJ20 44132013 EC50 = 1.585 nM T58921 CO7FK6 44132174 EC50 = 0.7943 nM T58921 C3ZW6T 44132175 EC50 = 0.5012 nM T58921 CAO4X6 44132177 EC50 = 125.89 nM T58921 C7ZA6G 44132181 EC50 = 15.85 nM T58921 CLW9Z0 44132339 EC50 = 0.5012 nM T58921 CEI15P 44132341 EC50 = 39.81 nM T58921 C42ZQI 44132343 EC50 = 794.33 nM T58921 C84BXQ 44132346 EC50 = 6.31 nM T58921 CUS7L8 44132498 EC50 = 50.12 nM T58921 CFC7O4 44132499 EC50 = 39.81 nM T58921 CTMK74 44132500 EC50 = 50.12 nM T58921 C8TJ3Y 44132501 EC50 = 630.96 nM T58921 CWY98Z 44132657 EC50 = 251.19 nM T58921 C9XSV8 44132658 EC50 = 125.89 nM T58921 C8AE7R 44132660 EC50 = 199.53 nM T58921 CVN3X4 44132816 EC50 = 398.11 nM T58921 C9F4JM 44132980 EC50 = 3.162 nM T58921 CF71RT 44133326 EC50 = 2.512 nM T58921 C9XAI6 44133327 EC50 = 79.43 nM T58921 C7MD4F 44133328 EC50 = 50.12 nM T58921 CL58XZ 44133329 EC50 = 79.43 nM T58921 CCFO06 44133330 EC50 = 31.62 nM T58921 CIKN25 44134057 EC50 = 501.19 nM T58921 CQ83EC 44143316 Ki = 2700 nM T58921 C12XUE 44143317 Ki = 300 nM T58921 CD2VC6 44143318 Ki = 5900 nM T58921 CBOX40 44143319 Ki = 2200 nM T58921 C1GQC6 44143320 Ki = 660 nM T58921 C9FRI3 44143321 Ki = 4100 nM T58921 C3DGV4 44143322 Ki = 5000 nM T58921 C0Z8NG 44143323 Ki = 7600 nM T58921 C6GJU8 44143324 Ki = 4000 nM T58921 CK25QY 44143325 EC50 > 10000 nM T58921 C9D6TL 44143326 Ki = 1200 nM T58921 C7U1JB 44143327 Ki = 77 nM T58921 C4OBI5 44143328 Ki = 84 nM T58921 C3ZL5T 44143329 Ki = 210 nM T58921 CX8Z3J 44143330 Ki = 43 nM T58921 CO72BR 44143331 Ki = 79 nM T58921 CZ3GO9 44143332 Ki = 20 nM T58921 C78CKO 44143333 Ki = 44 nM T58921 CLUG09 44143334 Ki = 25 nM T58921 C6VE7C 44143335 Ki = 30 nM T58921 CZF3A7 44143336 Ki = 170 nM T58921 C0UKO6 44143337 Ki = 39 nM T58921 CF2O9K 44143338 Ki = 150 nM T58921 CUG16K 44143339 Ki = 84 nM T58921 C4MB2X 44143340 Ki > 10000 nM T58921 C7BS4Z 44143341 Ki = 200 nM T58921 CNA0F7 44143342 Ki = 76 nM T58921 CM3N5P 44143343 Ki = 110 nM T58921 C5AK1N 44190592 EC50 = 1 nM T58921 CSN2I3 44190675 EC50 = 2 nM T58921 C7VP2C 44190676 IC50 = 17 nM T58921 C2AV1K 44190762 EC50 = 4 nM T58921 C2Z9AO 44190763 EC50 = 6 nM T58921 CT2VX9 44190764 EC50 = 1 nM T58921 C1HYW3 44190860 EC50 = 10 nM T58921 CGL02H 44190861 EC50 = 2 nM T58921 C2FIL5 44190862 EC50 = 2 nM T58921 C6MZ5G 44190863 EC50 = 2 nM T58921 CSE61I 44224204 EC50 = 20000000 nM T58921 CF29RT 44241498 EC50 = 398.11 nM T58921 COUQ71 44241499 EC50 = 572 nM T58921 C1B2ED 44246273 EC50 = 399 nM T58921 CMH0A5 44246274 EC50 = 65 nM T58921 CRE63N 44246275 EC50 > 20000 nM T58921 CLM3P2 44246276 EC50 > 20000 nM T58921 CON62P 44249904 EC50 = 3500 nM T58921 C98GDR 44249905 EC50 = 3900 nM T58921 C5LE2G 44263416 EC50 = 173 nM T58921 C46JLC 44263417 EC50 = 4500 nM T58921 CV24PU 44263418 EC50 = 9000 nM T58921 C63NTO 44263419 EC50 = 2000 nM T58921 CHV0U4 44263420 EC50 = 492 nM T58921 CST49K 44263421 EC50 = 2600 nM T58921 C2IV6K 44263422 EC50 = 3700 nM T58921 CB2L5E 44263423 EC50 = 2300 nM T58921 CJ8NG4 44263424 EC50 = 1200 nM T58921 CQF3S1 44263425 EC50 = 3600 nM T58921 CK0Y7P 44263426 EC50 = 480 nM T58921 CN8F7X 44263427 EC50 = 9000 nM T58921 CM4JU6 44263428 EC50 = 7000 nM T58921 C9ORI5 44263429 EC50 > 30000 nM T58921 C5A4HL 44273874 EC50 = 1400 nM T58921 CE58NO 44273875 EC50 = 10000 nM T58921 CMX75T 44273944 EC50 = 320 nM T58921 C0XNR5 44273963 EC50 = 1200 nM T58921 CC06QB 44273964 EC50 = 2000 nM T58921 CXOQ47 44274021 EC50 = 1000 nM T58921 CBY28T 44274044 EC50 = 1000 nM T58921 CNV3P0 44274047 EC50 = 2000 nM T58921 CH7M5T 44274107 EC50 = 1350 nM T58921 C67AKM 44316114 EC50 = 160 nM T58921 C1HKA2 44316347 EC50 = 79 nM T58921 CP3GE6 44316348 EC50 = 100 nM T58921 C27PUY 44316349 EC50 = 100 nM T58921 CJ4IP0 44316383 EC50 = 4 nM T58921 C1V6UE 44316496 EC50 = 16 nM T58921 CX1V8Q 44316506 EC50 = 50 nM T58921 CX07YR 44316521 EC50 = 20 nM T58921 C1LBQ7 44316568 EC50 = 100 nM T58921 CI19KT 44316591 EC50 = 63 nM T58921 CNG0H5 44316592 EC50 = 25 nM T58921 CDPY05 44316628 EC50 = 25 nM T58921 CXC9R4 44316629 EC50 = 40 nM T58921 C64ETY 44316824 EC50 = 32 nM T58921 CLQ0B3 44316825 EC50 = 2 nM T58921 CD2HP8 44316826 EC50 = 13 nM T58921 C29KBV 44316844 EC50 = 230 nM T58921 CKC5F4 44316880 EC50 = 6 nM T58921 CFT53Z 44316903 EC50 = 4 nM T58921 C3E7QU 44320897 EC50 = 1500 nM T58921 CIY30P 44320978 EC50 = 600 nM T58921 C6J0GY 44321201 EC50 = 3981.07 nM T58921 CLBK38 44321284 EC50 = 800 nM T58921 C4IR1A 44321440 EC50 = 2691.53 nM T58921 C45WMS 44321441 EC50 = 4265.8 nM T58921 CR3T1Q 44321462 EC50 = 2000 nM T58921 C9AEI4 44321463 EC50 = 2187.76 nM T58921 CRFU18 44321490 EC50 = 2900 nM T58921 CQ10AI 44321517 EC50 = 3300 nM T58921 CH6Z2D 44321548 EC50 = 1698.24 nM T58921 C6ZK4E 44321572 EC50 = 590 nM T58921 CQ3RA9 44321573 EC50 = 3090.3 nM T58921 C6HM2Z 44321655 EC50 = 8500 nM T58921 CH1U9W 44323732 EC50 = 36000 nM T58921 C8N7LP 44331667 EC50 = 320 nM T58921 CRG71X 44331668 EC50 = 30 nM T58921 CR9E3N 44331685 EC50 = 0.5 nM T58921 CTFW53 44331750 EC50 = 170 nM T58921 CRNL38 44331751 EC50 = 81 nM T58921 CKWC85 44335916 Ki = 620 nM T58921 COF23R 44335940 Ki = 360 nM T58921 CQHJ92 44335944 EC50 = 23.99 nM T58921 C46TRE 44335970 EC50 = 138 nM T58921 C0SYL4 44335992 EC50 = 410 nM T58921 C9M2TC 44335993 Ki = 280 nM T58921 CY1L8T 44336013 Ki = 2600 nM T58921 C4S9KU 44336048 Ki = 2100 nM T58921 CW8E2Z 44336264 EC50 = 710 nM T58921 CI9AN1 44337634 Ki > 10000 nM T58921 CR9YS1 44337635 Ki = 8530 nM T58921 CRA5F6 44337688 Ki = 79 nM T58921 CEMT31 44337693 Ki = 4600 nM T58921 CZ7J0I 44337694 Ki = 194 nM T58921 CL1HK2 44337695 Ki = 3149 nM T58921 C4X6LA 44337716 Ki = 5940 nM T58921 CCQ67S 44337866 Ki = 110 nM T58921 CRJ87P 44338182 Ki = 985 nM T58921 CWB32K 44338195 Ki = 560 nM T58921 CA36CR 44339522 EC50 = 80 nM T58921 CV3R2S 44339547 IC50 = 1400 nM T58921 C4EW3V 44341104 Ki = 213.8 nM T58921 C97XPN 44341140 Ki = 549.54 nM T58921 CZ24RC 44341151 Ki = 1905.46 nM T58921 CC30FI 44341152 Ki < 10000 nM T58921 CVC1Q6 44341153 Ki = 4466.84 nM T58921 CT0DS3 44341159 EC50 < 10000 nM T58921 C98PGA 44341160 EC50 = 3019.95 nM T58921 CZM5S1 44341161 Ki < 10000 nM T58921 C4F8KD 44341362 EC50 = 338.84 nM T58921 CZ25OL 44344272 EC50 = 3800 nM T58921 C9C8FN 44344313 EC50 = 3160 nM T58921 CWD8B7 44344585 EC50 = 2880 nM T58921 CMC41U 44345158 Ki = 160 nM T58921 C4MTA7 44345159 Ki = 170 nM T58921 CR0GI8 44345164 Ki = 100 nM T58921 CR7EX2 44345170 Ki = 180 nM T58921 CX2I7F 44345171 Ki = 1400 nM T58921 CH9F6O 44345180 EC50 = 300 nM T58921 CXY46J 44345202 EC50 = 300 nM T58921 CU7F4O 44345203 Ki = 600 nM T58921 CC3FJ0 44345204 EC50 = 700 nM T58921 CMR75E 44345354 EC50 = 700 nM T58921 C5WY9X 44345355 EC50 = 300 nM T58921 CANH09 44345363 EC50 = 700 nM T58921 CPHO86 44345406 Ki = 500 nM T58921 C2FGP1 44345407 EC50 = 600 nM T58921 C2BKP7 44345432 Ki = 1500 nM T58921 CY7O8G 44345843 EC50 = 2500 nM T58921 C0CS9D 44348875 EC50 = 1600 nM T58921 CG6H2T 44353335 EC50 = 7.4 nM T58921 CW0T6K 44353336 EC50 = 4.7 nM T58921 C8K0AB 44353347 EC50 = 4.1 nM T58921 C3DYE9 44353422 EC50 = 0.8 nM T58921 C5DTY3 44353441 EC50 = 2.7 nM T58921 C2M8TN 44353456 EC50 = 15.1 nM T58921 CVKA40 44353466 EC50 = 16.3 nM T58921 C8J5SA 44353480 EC50 = 2.7 nM T58921 CIB15X 44353481 EC50 = 0.7 nM T58921 CQS0E8 44364361 Ki = 1258.93 nM T58921 C3E9FH 44364377 Ki < 3162.28 nM T58921 CXUP19 44364423 EC50 = 446.68 nM T58921 C8MG3C 44364499 Ki = 28.18 nM T58921 C32PRI 44364575 Ki = 162.18 nM T58921 C2UM3P 44364622 Ki < 3162.28 nM T58921 C8ZPF2 44364623 Ki < 3162.28 nM T58921 CMKB89 44364633 Ki < 3162.28 nM T58921 CQ0F2H 44364634 Ki < 3162.28 nM T58921 CZB1E8 44364682 EC50 = 0.302 nM T58921 CW8M2A 44364691 EC50 = 0.4266 nM T58921 CB74RL 44364769 Ki = 4.169 nM T58921 C2JVP4 44364787 EC50 = 0.5754 nM T58921 C9K5MW 44364872 Ki = 645.65 nM T58921 C5IE3N 44364876 Ki = 11.48 nM T58921 CAR27T 44364953 EC50 = 208.93 nM T58921 CS3C7W 44365532 IC50 = 6100 nM T58921 CM1X4H 44379496 EC50 = 12400 nM T58921 CZ5BG6 44383664 Ki = 26 nM T58921 CK9PD5 44383828 Ki = 20 nM T58921 CIVC76 44383831 EC50 = 37 nM T58921 CMB3S2 44383889 Ki = 8.9 nM T58921 C5ND3Y 44384224 Ki > 5300 nM T58921 CW9LD2 44384226 EC50 = 10 nM T58921 CPY0K6 44384403 Ki = 616 nM T58921 CD4KM5 44384407 Ki = 152 nM T58921 C53DOZ 44384408 Ki = 1330 nM T58921 CTJD81 44384415 Ki = 662 nM T58921 CKDS82 44384419 EC50 = 2 nM T58921 CA7YK9 44384460 Ki = 13 nM T58921 C4W7VN 44384466 Ki = 348 nM T58921 C46RVE 44384539 Ki = 52 nM T58921 C6PIU9 44384589 EC50 = 16 nM T58921 C4R6EW 44384639 Ki = 22 nM T58921 CM8AE6 44385177 Ki = 498 nM T58921 C2FQX7 44385248 Ki = 100 nM T58921 CFM56P 44385352 Ki = 115 nM T58921 CE47ZL 44385396 Ki = 41 nM T58921 C6H0OL 44385399 Ki = 448 nM T58921 CY2O5S 44385405 Ki = 304 nM T58921 CH9UP4 44385406 Ki = 145 nM T58921 CRWI98 44386508 EC50 = 4 nM T58921 CDN54E 44388167 EC50 = 3000 nM T58921 C50FPR 44388210 EC50 = 1000 nM T58921 C5DNU7 44388563 EC50 = 500 nM T58921 C51XZF 44388650 IC50 > 15000 nM T58921 C8E1NU 44388684 IC50 > 15000 nM T58921 CA1XK7 44388810 IC50 > 15000 nM T58921 CU1Y8L 44388819 IC50 > 15000 nM T58921 CU71OL 44388848 EC50 = 1000 nM T58921 C28TPK 44388866 EC50 = 3000 nM T58921 CMQ25R 44388882 IC50 > 15000 nM T58921 CQ6Z4Y 44388907 EC50 = 700 nM T58921 CBV25F 44388914 IC50 = 15000 nM T58921 C57OKZ 44388945 IC50 = 4690 nM T58921 C0EH5G 44388966 EC50 = 2 nM T58921 CF7L8V 44388968 EC50 = 1000 nM T58921 CH0TL9 44388998 EC50 = 6 nM T58921 C9FQ1S 44389035 EC50 = 280 nM T58921 C5V0PS 44389085 EC50 = 3 nM T58921 C0S6QK 44389098 EC50 = 2 nM T58921 C6GF3L 44389191 EC50 = 240 nM T58921 COXA71 44389801 EC50 = 8000 nM T58921 C9Q2GR 44391841 IC50 = 6280 nM T58921 C78VSM 44392315 EC50 = 305 nM T58921 C83DZJ 44396236 EC50 = 4 nM T58921 CDC15W 44399773 IC50 = 29 nM T58921 CZO8C3 44399778 EC50 = 3 nM T58921 C29NJR 44399829 IC50 = 466 nM T58921 C58CAS 44399878 IC50 = 135 nM T58921 CV08EP 44399967 EC50 = 31 nM T58921 CJ0DB4 44399972 EC50 = 39 nM T58921 CW3AX4 44399983 IC50 = 2 nM T58921 C0B8IW 44400079 IC50 = 641 nM T58921 CT09WZ 44400131 EC50 = 16 nM T58921 C60YCL 44404190 IC50 = 3900 nM T58921 C21HNW 44404248 Ki > 10000 nM T58921 CD79BV 44404256 Ki > 10000 nM T58921 CMQI41 44404263 EC50 = 1413 nM T58921 C6G1EF 44404267 Ki = 718 nM T58921 CGX5M8 44404271 Ki = 579 nM T58921 CICB09 44404275 Ki > 10000 nM T58921 CGD96V 44404636 IC50 = 21 nM T58921 C5F9ZX 44404637 EC50 = 299 nM T58921 CQ9V3L 44404648 IC50 = 104 nM T58921 CL3OB9 44404649 IC50 = 202 nM T58921 C6EIY9 44404654 IC50 = 58 nM T58921 CR59YU 44404675 IC50 = 49 nM T58921 CZ53YS 44404680 IC50 = 49 nM T58921 CUX13J 44404681 IC50 = 78 nM T58921 C6D7SO 44404685 IC50 = 115 nM T58921 CUX92K 44404686 IC50 = 107 nM T58921 C4TQ6X 44404690 IC50 = 60 nM T58921 CY35ZW 44404691 IC50 = 120 nM T58921 C8RPC4 44404696 IC50 = 102 nM T58921 C7Z5ST 44404700 IC50 = 298 nM T58921 C5IUA7 44404701 EC50 = 106 nM T58921 CS8NO5 44404703 IC50 = 19 nM T58921 CL30JV 44404704 IC50 = 17 nM T58921 C7GNI4 44404708 IC50 = 83 nM T58921 C48RBM 44404714 IC50 = 13 nM T58921 CJH5X6 44404715 IC50 = 39 nM T58921 CHNT04 44404717 IC50 = 318 nM T58921 C7ZSM1 44404718 EC50 = 34 nM T58921 CT15BE 44404723 IC50 = 18 nM T58921 C3UB2D 44404727 EC50 = 126 nM T58921 C5GZP7 44404728 IC50 = 5 nM T58921 COI8L9 44404729 EC50 = 2 nM T58921 CM96VZ 44404734 IC50 = 75 nM T58921 CP7U3J 44404735 EC50 = 34 nM T58921 C7IJ5H 44405121 EC50 = 1810 nM T58921 CFZB63 44406104 EC50 = 523 nM T58921 CDAF49 44406106 EC50 = 153 nM T58921 CDA3Z9 44406117 EC50 = 396 nM T58921 CJ7F5L 44406154 EC50 = 330 nM T58921 CC0Y3J 44406172 EC50 = 49 nM T58921 CS06AB 44406180 EC50 = 247 nM T58921 CA1XV3 44406204 EC50 = 77 nM T58921 CB1X2D 44406205 EC50 = 84 nM T58921 C7AD9N 44406236 EC50 = 368 nM T58921 CB0E4H 44406258 EC50 > 10000 nM T58921 CI47RY 44406262 EC50 = 632 nM T58921 CSO0P7 44406263 EC50 > 10000 nM T58921 C95DYP 44406265 EC50 = 738 nM T58921 C2XDJ1 44406266 EC50 = 94 nM T58921 C7K6HJ 44406267 EC50 > 10000 nM T58921 C3I0MQ 44406283 EC50 = 9560 nM T58921 CK4Z7J 44406288 EC50 > 10000 nM T58921 CXY5J2 44406292 EC50 = 43 nM T58921 CUW97K 44406303 EC50 > 10000 nM T58921 C6KL7U 44406304 EC50 > 10000 nM T58921 CA91XP 44406318 EC50 > 10000 nM T58921 CPN2F1 44406331 EC50 = 5640 nM T58921 C13MXB 44406336 EC50 = 177 nM T58921 C9GNW2 44406340 EC50 = 85 nM T58921 CT4Z8O 44406341 EC50 > 10000 nM T58921 CB6S1C 44406344 EC50 = 196 nM T58921 C0WAS9 44406345 EC50 > 10000 nM T58921 CRY47S 44406364 EC50 > 10000 nM T58921 C5U1OQ 44406365 EC50 > 10000 nM T58921 C3KIO7 44406367 EC50 = 45 nM T58921 CQ20JM 44406375 EC50 > 10000 nM T58921 CK10VQ 44406381 EC50 = 46 nM T58921 C1WPX7 44406411 EC50 = 83 nM T58921 C4IBL1 44406437 EC50 = 160 nM T58921 CV5L8T 44406441 EC50 > 10000 nM T58921 C7R5NB 44406455 EC50 = 225 nM T58921 C2Z7XC 44406472 EC50 = 605 nM T58921 CKA1Z0 44406477 EC50 = 6 nM T58921 C1OFD9 44406482 EC50 = 46 nM T58921 C4IOC7 44406528 EC50 = 762 nM T58921 CW70MB 44406532 EC50 = 19 nM T58921 C0Y4EZ 44406533 EC50 = 95 nM T58921 CDX97W 44407180 EC50 > 10000 nM T58921 CU24FD 44407220 EC50 = 500 nM T58921 CJO4I9 44407221 EC50 = 1600 nM T58921 C7X4UM 44407224 EC50 > 10000 nM T58921 CD7W9V 44409035 EC50 > 3000 nM T58921 C3I7OD 44409044 IC50 = 981 nM T58921 CTA6G7 44409088 EC50 = 1087 nM T58921 C6TRF5 44409127 EC50 > 3000 nM T58921 CJ8A6M 44409131 IC50 = 851 nM T58921 C6Y1XC 44409170 IC50 = 6440 nM T58921 CB02UG 44409181 EC50 = 7690 nM T58921 C7FMA5 44409249 IC50 = 1851 nM T58921 CAN69Y 44409279 IC50 > 6000 nM T58921 C76RXA 44409375 IC50 = 3610 nM T58921 C3ODA1 44409427 IC50 = 1240 nM T58921 CU30EB 44411547 EC50 > 10000 nM T58921 CYER28 44411548 EC50 > 10000 nM T58921 CBYE57 44411557 EC50 > 10000 nM T58921 CWR6V3 44411558 EC50 > 10000 nM T58921 C5IWC6 44411561 EC50 > 10000 nM T58921 C8G1HJ 44411562 EC50 > 10000 nM T58921 CNO49B 44411563 EC50 > 10000 nM T58921 C25NTU 44411565 EC50 > 10000 nM T58921 C3G2CA 44411571 EC50 > 10000 nM T58921 C4W6DO 44411577 EC50 > 10000 nM T58921 CFB63G 44411578 EC50 > 10000 nM T58921 CM0RU6 44411581 EC50 > 10000 nM T58921 COB80S 44411616 EC50 > 10000 nM T58921 C4C9LD 44411618 EC50 > 10000 nM T58921 CY8K9S 44411630 EC50 > 10000 nM T58921 CNL81R 44411653 IC50 = 279.9 nM T58921 CW3AV8 44411661 IC50 = 270 nM T58921 C5P4BM 44411708 EC50 > 10000 nM T58921 C5AR4E 44411737 EC50 > 10000 nM T58921 C06BPM 44411740 EC50 > 10000 nM T58921 C2G1LB 44411741 EC50 > 10000 nM T58921 CQL2Z4 44411767 EC50 > 10000 nM T58921 C2KCO7 44411772 EC50 > 10000 nM T58921 C4U2SJ 44411842 IC50 = 2897.34 nM T58921 CJF9L1 44411843 IC50 = 102 nM T58921 CV3N5O 44411918 EC50 = 1200 nM T58921 CFU5X3 44411943 EC50 > 10000 nM T58921 CP1AZ6 44411945 EC50 = 370 nM T58921 C70NKQ 44411946 EC50 = 740 nM T58921 C71ZSM 44411968 EC50 > 10000 nM T58921 CX6DN0 44411977 IC50 = 2999.16 nM T58921 C8DPK5 44412188 IC50 = 460 nM T58921 CPK6G2 44412195 IC50 = 4600 nM T58921 CNVG17 44413626 EC50 = 28000 nM T58921 CDTM49 44413635 EC50 = 11050 nM T58921 C1GH3B 44414891 EC50 > 10000 nM T58921 CU8NQ5 44414900 EC50 > 10000 nM T58921 CKM0I8 44414901 EC50 > 10000 nM T58921 C7LCH5 44414917 EC50 > 10000 nM T58921 CBQ62J 44414926 EC50 > 10000 nM T58921 C07VTH 44414927 EC50 = 3230 nM T58921 C1ETO8 44414955 EC50 > 10000 nM T58921 CV8IA5 44414956 EC50 > 10000 nM T58921 CTK8Z0 44414962 EC50 > 10000 nM T58921 C1G4OC 44414967 EC50 > 10000 nM T58921 C64UOB 44414968 EC50 > 10000 nM T58921 CLO83A 44414991 EC50 > 10000 nM T58921 C23ARN 44415004 EC50 = 1250 nM T58921 C0TI2L 44415602 EC50 = 1261 nM T58921 C4ZDC7 44415616 EC50 = 153 nM T58921 C04EOY 44415664 EC50 = 288 nM T58921 C1UO6R 44415696 EC50 = 757 nM T58921 C6C0YB 44415715 EC50 = 1185 nM T58921 C9NB7J 44419009 EC50 > 10000 nM T58921 C97QXT 44419013 EC50 > 10000 nM T58921 C4P1SD 44419253 IC50 = 60 nM T58921 C4B1HD 44419255 IC50 = 1 nM T58921 C3QXT5 44419348 IC50 = 720 nM T58921 C1BE0F 44419349 IC50 = 280 nM T58921 CP51GU 44419352 IC50 = 80 nM T58921 CL8S2O 44419353 IC50 = 290 nM T58921 C9HR0J 44419354 IC50 = 180 nM T58921 C92YZG 44419355 IC50 = 90 nM T58921 C3YC9M 44419356 IC50 = 80 nM T58921 C7F0QG 44419357 IC50 = 80 nM T58921 C6KLM0 44419361 IC50 = 680 nM T58921 CCA39P 44419362 IC50 = 700 nM T58921 CJD4H7 44419365 IC50 = 140 nM T58921 CTK13E 44419366 IC50 = 90 nM T58921 C6OKQ3 44419369 IC50 = 9400 nM T58921 CVX86S 44419372 IC50 = 2440 nM T58921 CP4T6W 44419373 IC50 = 400 nM T58921 CNY83B 44419381 IC50 = 50 nM T58921 C9ERV0 44419382 IC50 = 280 nM T58921 CA5L1Q 44419383 IC50 = 770 nM T58921 CIXL31 44419385 IC50 = 380 nM T58921 CW9SG8 44419386 IC50 = 330 nM T58921 CSD0I4 44419387 IC50 = 330 nM T58921 CV9TL4 44419389 IC50 = 540 nM T58921 C1XM7I 44419390 IC50 = 7 nM T58921 C8H5TX 44419391 IC50 = 7 nM T58921 CMT5G1 44419392 IC50 = 2 nM T58921 CUZ7L4 44419393 IC50 = 290 nM T58921 CP0F9T 44419760 EC50 = 5 nM T58921 CBZ5D8 44419765 EC50 = 1280 nM T58921 CC6U1K 44419769 Ki = 360 nM T58921 C17UJG 44419770 Ki = 12000 nM T58921 C2A5CS 44419772 EC50 = 28 nM T58921 C0J5VZ 44419773 EC50 = 984 nM T58921 CCA53N 44419776 EC50 = 6 nM T58921 CF6E9L 44419778 Ki = 15 nM T58921 CT8CU5 44419780 EC50 = 2810 nM T58921 CWK6C9 44419783 Ki = 73 nM T58921 CL74CP 44419785 EC50 = 1010 nM T58921 C6Z9KE 44419786 EC50 = 125 nM T58921 CUQJ29 44419790 Ki = 3500 nM T58921 C3K6RF 44419795 Ki = 6 nM T58921 CUW52F 44419799 Ki = 17000 nM T58921 C39JPK 44419805 Ki = 810 nM T58921 CM2YG0 44419807 Ki = 1100 nM T58921 C8E6CZ 44419808 EC50 = 22 nM T58921 C2ABF5 44419809 EC50 = 5 nM T58921 C7XB3Q 44419814 EC50 = 42 nM T58921 CKOR70 44419819 EC50 = 6 nM T58921 C03BNV 44419822 EC50 = 268 nM T58921 CNX3V9 44419827 EC50 = 65 nM T58921 CN62LT 44419828 Ki = 240 nM T58921 CT8OY2 44419830 Ki = 15 nM T58921 CY60PA 44419884 EC50 = 887 nM T58921 CH8RG7 44419890 Ki = 93 nM T58921 CP8OT7 44419891 EC50 = 130 nM T58921 C7XY6Z 44419898 EC50 = 5 nM T58921 C9FXY7 44419906 EC50 = 12 nM T58921 CY2QX8 44419911 Ki = 2300 nM T58921 CC7PF3 44419918 EC50 > 10000 nM T58921 CCI9O8 44419924 EC50 = 26 nM T58921 C9ZP8B 44420402 EC50 = 9 nM T58921 C4HR6P 44420473 EC50 = 2684 nM T58921 CL9N8S 44420479 IC50 = 161 nM T58921 C5IQ7K 44420484 IC50 = 72 nM T58921 CZ67XE 44420485 EC50 = 2 nM T58921 C5QOU1 44420506 EC50 = 7 nM T58921 CBWX49 44420565 EC50 = 77 nM T58921 C72TSL 44420566 EC50 = 8 nM T58921 CL86VI 44424582 EC50 = 1800 nM T58921 CV8X0N 44424583 EC50 = 1300 nM T58921 C4QN7D 44424584 EC50 = 6200 nM T58921 CK89CE 44424585 EC50 = 2200 nM T58921 CNS39L 44424586 EC50 = 650 nM T58921 CGCJ17 44424587 EC50 = 1400 nM T58921 C6LXQ5 44424588 EC50 = 7000 nM T58921 CBZ1C3 44424589 EC50 > 10000 nM T58921 CBZU45 44424590 EC50 > 10000 nM T58921 CC32AV 44424591 EC50 = 3600 nM T58921 CQ1KL3 44424592 EC50 = 2400 nM T58921 CG1CE6 44424593 EC50 = 1500 nM T58921 CL2K0C 44424594 EC50 = 1000 nM T58921 CSGM27 44424595 EC50 = 1000 nM T58921 C62FYL 44425829 Ki = 100 nM T58921 CZ2L7O 44425831 Ki = 112.2 nM T58921 C4G1PR 44425833 Ki = 158.49 nM T58921 CWC2Q6 44425836 Ki = 173.78 nM T58921 C4CW7J 44425838 Ki = 309.03 nM T58921 C4AEB5 44425840 Ki = 51.29 nM T58921 C2MW7R 44425841 Ki = 165.96 nM T58921 CFG86S 44425842 Ki = 194.98 nM T58921 CR6QK9 44425843 Ki = 114.82 nM T58921 CZBM48 44425844 Ki = 144.54 nM T58921 C7PBD8 44425845 Ki = 269.15 nM T58921 CBFM17 44425846 Ki = 47.86 nM T58921 CP0Q3K 44425847 Ki = 61.66 nM T58921 CQV40O 44425848 Ki = 87.1 nM T58921 C30EJO 44425850 EC50 > 1000 nM T58921 CQ9RH6 44425851 EC50 > 1000 nM T58921 CH13TY 44425852 EC50 > 1000 nM T58921 CGE39L 44425853 EC50 > 1000 nM T58921 CX39CR 44425854 EC50 > 1000 nM T58921 CBJU72 44425855 EC50 > 1000 nM T58921 C3QLV7 44425856 EC50 > 1000 nM T58921 CZ3X6Y 44425859 EC50 > 1000 nM T58921 CN8A9Y 44425862 EC50 > 1000 nM T58921 CP7JN9 44425864 EC50 > 1000 nM T58921 CP6SO9 44425869 EC50 > 1000 nM T58921 CDVH71 44425872 EC50 > 1000 nM T58921 CI0Q3G 44431866 EC50 = 350 nM T58921 CYIK84 44431867 EC50 = 580 nM T58921 C6C0VT 44431868 EC50 = 4580 nM T58921 COF38E 44431869 EC50 = 1050 nM T58921 C8QW9M 44431873 EC50 = 490 nM T58921 C9MRU3 44431876 EC50 = 140 nM T58921 CX5QL8 44431880 EC50 = 5390 nM T58921 CC81BQ 44431882 EC50 = 3480 nM T58921 CVHO05 44431883 EC50 = 3600 nM T58921 CZ9RU5 44431884 EC50 = 1060 nM T58921 C05BKW 44431885 EC50 = 1420 nM T58921 C86NSF 44431886 EC50 = 1400 nM T58921 CAPN49 44431887 EC50 = 7170 nM T58921 C06KRB 44432398 IC50 = 6260 nM T58921 CWDS06 44432399 IC50 > 10000 nM T58921 C9YZ1I 44432400 IC50 > 10000 nM T58921 CK6PU9 44432401 IC50 = 7580 nM T58921 CSF09X 44432402 IC50 = 5790 nM T58921 CE51LN 44432403 IC50 = 3730 nM T58921 CDV5O8 44432404 IC50 > 10000 nM T58921 CN7KJ9 44432405 IC50 = 5395.11 nM T58921 CMO9I5 44432406 IC50 > 10000 nM T58921 CA7OU6 44432407 IC50 > 10000 nM T58921 C12ANM 44432408 IC50 > 10000 nM T58921 CQ1W3L 44432409 IC50 > 10000 nM T58921 C8AQ3I 44432410 IC50 > 10000 nM T58921 CJ7GY1 44432411 IC50 > 10000 nM T58921 CI45BS 44432832 EC50 > 10000 nM T58921 CRPF69 44432835 EC50 > 10000 nM T58921 C0BO8H 44432848 EC50 > 10000 nM T58921 C5C4HV 44432849 EC50 > 10000 nM T58921 C2D5YP 44432852 EC50 > 10000 nM T58921 CBC74Q 44432853 EC50 > 10000 nM T58921 C1A9NX 44432854 EC50 > 10000 nM T58921 CF3L8X 44432855 EC50 = 6600 nM T58921 C9ETG7 44432856 EC50 > 10000 nM T58921 CWF49O 44434337 IC50 = 18 nM T58921 C53YEQ 44434338 EC50 = 57 nM T58921 C74NKE 44434339 EC50 = 49 nM T58921 C43PNF 44434340 IC50 = 12 nM T58921 CGD7Q8 44434341 EC50 = 43 nM T58921 CQP74N 44434342 IC50 = 203 nM T58921 CVWA23 44434343 IC50 = 114 nM T58921 C0VAZ9 44434344 IC50 = 7 nM T58921 C5WY9B 44434345 IC50 = 6.998 nM T58921 CM4K1D 44434346 EC50 = 28 nM T58921 CKI70B 44434347 EC50 = 10 nM T58921 CH5JP2 44434348 EC50 = 26 nM T58921 CQW7J6 44434349 EC50 = 125 nM T58921 CS31PG 44434350 IC50 = 5 nM T58921 CERT39 44434351 IC50 = 16.98 nM T58921 C4B8VJ 44434352 EC50 = 22 nM T58921 CM8VY6 44434353 IC50 = 7.998 nM T58921 C9IG2C 44434354 EC50 = 1088 nM T58921 C4SMI1 44434355 IC50 = 13 nM T58921 C3O2BF 44434356 IC50 = 233 nM T58921 CRBM37 44434357 EC50 = 32 nM T58921 CL2H8U 44434358 IC50 = 36.98 nM T58921 CB5U3S 44434359 IC50 = 95.06 nM T58921 C4K0FY 44434360 EC50 = 135 nM T58921 CIA86O 44434361 EC50 = 24 nM T58921 C2VG9W 44434362 EC50 = 163 nM T58921 CL5AH3 44439623 IC50 = 567.54 nM T58921 CF01IC 44439624 IC50 = 1088.93 nM T58921 C64AHD 44439625 EC50 = 2300 nM T58921 CIW8B5 44439626 EC50 = 140 nM T58921 C7YHU2 44439631 EC50 = 2270 nM T58921 CL1XI5 44439632 IC50 = 979 nM T58921 CM6Q0Y 44439633 IC50 = 20 nM T58921 C1JAZ3 44440776 EC50 = 1000 nM T58921 CYOD04 44440777 EC50 = 1100 nM T58921 CIR27Y 44440779 EC50 = 530 nM T58921 CG43HK 44440780 EC50 = 400 nM T58921 CNI45S 44440781 EC50 > 10000 nM T58921 CQ25AW 44440782 EC50 = 1600 nM T58921 CWO5C2 44440783 EC50 = 2000 nM T58921 C3-OCT 44440785 EC50 > 10000 nM T58921 C6TMR4 44440786 EC50 = 1800 nM T58921 C03TVK 44440787 EC50 > 10000 nM T58921 C1V0CH 44440788 EC50 > 10000 nM T58921 C4NDM7 44440789 EC50 = 210 nM T58921 COI23R 44440790 EC50 = 130 nM T58921 C8TOE9 44440791 EC50 = 750 nM T58921 C4BQ1C 44440792 EC50 = 2100 nM T58921 CDZ45N 44440795 EC50 = 1800 nM T58921 CA7G3R 44440797 EC50 = 1400 nM T58921 C1PQ7V 44440800 EC50 = 910 nM T58921 CX3P1C 44440804 EC50 = 870 nM T58921 C62VTF 44440805 EC50 = 940 nM T58921 CWDC32 44440806 EC50 = 1190 nM T58921 CRS8Z5 44440928 EC50 = 6340 nM T58921 C9F4ME 44440929 EC50 = 3690 nM T58921 CUJ8X0 44441213 EC50 = 4100 nM T58921 CRWN48 44441214 EC50 = 1200 nM T58921 CV6RK5 44441215 EC50 = 200 nM T58921 CQ23GJ 44441216 EC50 = 80 nM T58921 CX5M7Q 44441220 EC50 = 190 nM T58921 CY74RZ 44441221 EC50 = 3100 nM T58921 C3AS9D 44441223 EC50 = 3000 nM T58921 CBY9C7 44441224 EC50 = 5100 nM T58921 CEP16Z 44441344 EC50 = 300 nM T58921 CTE95F 44441446 EC50 = 108 nM T58921 C8YB9P 44441447 IC50 = 773 nM T58921 C7M2GD 44441451 IC50 = 183 nM T58921 CZ41WB 44441453 EC50 = 1390 nM T58921 C3FJM9 44441455 IC50 = 540 nM T58921 CY64MC 44441459 EC50 = 136 nM T58921 CH28FD 44441461 EC50 = 1800 nM T58921 CS9OP6 44441462 EC50 = 1180 nM T58921 C0RAC7 44441463 EC50 = 307 nM T58921 CBTE20 44441464 EC50 = 391 nM T58921 C06SRV 44441466 EC50 = 221 nM T58921 C9TRS0 44441467 EC50 = 840 nM T58921 CM1HQ6 44441469 EC50 = 230 nM T58921 C19DQE 44442440 EC50 = 3140 nM T58921 C2YD9E 44442441 EC50 = 14 nM T58921 C1APG0 44442442 EC50 = 3 nM T58921 C6RVT7 44442443 EC50 = 18 nM T58921 CAW91Q 44442444 EC50 = 3 nM T58921 CT68PM 44442445 EC50 = 21 nM T58921 C0IGW2 44442446 EC50 = 1 nM T58921 C8A6SM 44442447 EC50 = 13 nM T58921 CPFJ29 44442448 EC50 = 7 nM T58921 CF3D6P 44442449 EC50 = 64 nM T58921 CMQ17O 44442450 EC50 = 3 nM T58921 CL4K7X 44442451 EC50 = 11 nM T58921 CGCN21 44442452 EC50 = 0.8 nM T58921 CM1PL8 44442453 EC50 = 61 nM T58921 CORC37 44442454 EC50 = 7 nM T58921 C13HNY 44442455 EC50 = 47 nM T58921 C16NTG 44442456 EC50 = 116 nM T58921 C31ZGW 44442457 EC50 = 1.5 nM T58921 CLJ21W 44442458 EC50 = 30 nM T58921 CN14PT 44442459 EC50 = 272 nM T58921 CY1BJ8 44442460 EC50 = 30 nM T58921 C9EB3R 44442461 EC50 = 2 nM T58921 CO3GE5 44442462 EC50 = 13 nM T58921 CJ14GS 44442463 EC50 = 28 nM T58921 CEQB08 44442464 EC50 = 309 nM T58921 CYZA32 44442465 EC50 = 31 nM T58921 C3LA4I 44442466 EC50 = 347 nM T58921 C5VRE4 44442467 EC50 = 86 nM T58921 CYUR21 44442468 EC50 = 10000 nM T58921 CM6IW4 44442469 EC50 = 257 nM T58921 CORA57 44442470 EC50 = 10000 nM T58921 CA7MO3 44442471 EC50 = 7 nM T58921 CU0H8W 44442472 EC50 = 5 nM T58921 C6M0JQ 44442473 EC50 = 11 nM T58921 CH8SN0 44442474 EC50 = 10 nM T58921 C37QUO 44442475 EC50 = 607 nM T58921 CHIA45 44443517 EC50 = 1500 nM T58921 CWGR41 44443520 EC50 > 10000 nM T58921 CQJ8K0 44443529 EC50 = 150 nM T58921 CK5W0P 44443530 EC50 = 190 nM T58921 CSJ95Q 44443534 EC50 > 1000 nM T58921 CIQ4U0 44443538 EC50 = 70 nM T58921 CAWY35 44443563 EC50 = 150 nM T58921 C31WIL 44446245 EC50 > 10000 nM T58921 CI64WZ 44446247 EC50 > 10000 nM T58921 C6XIU3 44446250 EC50 > 10000 nM T58921 CHY27Q 44446252 EC50 > 10000 nM T58921 CE1S5F 44446255 EC50 > 10000 nM T58921 C9OGX2 44446257 EC50 > 10000 nM T58921 CI49YJ 44446258 EC50 > 10000 nM T58921 CSH1U8 44446260 EC50 = 5500 nM T58921 C7YSZ5 44446262 EC50 = 500 nM T58921 C9GMW7 44446263 EC50 = 300 nM T58921 CIR02A 44446264 EC50 > 10000 nM T58921 C3T2VM 44447156 Ki = 10000 nM T58921 CEJV01 44447159 Ki = 10000 nM T58921 CI97LH 44447160 Ki = 10000 nM T58921 CUL81F 44447162 Ki = 48 nM T58921 C4QYL8 44447163 Ki = 89 nM T58921 C5TKE9 44448345 IC50 > 25000 nM T58921 CI6HR5 44448403 IC50 > 25000 nM T58921 CTH06F 44448484 IC50 > 15000 nM T58921 C3DO6H 44448487 IC50 > 20000 nM T58921 C4KSB3 44448593 IC50 > 15000 nM T58921 CE29ID 44448632 IC50 > 15000 nM T58921 CE09DJ 44448767 EC50 = 28 nM T58921 C1NX8Y 44448801 EC50 = 5570 nM T58921 CRK9D8 44449001 EC50 = 8 nM T58921 C4HAK6 44449024 EC50 = 16 nM T58921 CW3BX7 44449049 EC50 = 40 nM T58921 CR94MO 44449074 EC50 = 4920 nM T58921 CC90BY 44449076 EC50 = 89 nM T58921 C8DS6T 44449100 EC50 = 170 nM T58921 CX0FP8 44449101 EC50 = 580 nM T58921 CF8U1H 44449125 EC50 = 6 nM T58921 CD1Q7S 44449127 EC50 = 18 nM T58921 CW9YO3 44449128 EC50 = 209 nM T58921 C1E5UC 44449161 EC50 = 44 nM T58921 C9P7JK 44449163 EC50 = 5 nM T58921 CP54JF 44449192 EC50 = 235 nM T58921 CR1W3G 44449220 EC50 > 7500 nM T58921 C85TKY 44451190 EC50 > 3000 nM T58921 CUM0J1 44453644 IC50 = 3400 nM T58921 CX46EF 44453670 EC50 = 840 nM T58921 CXPD58 44453913 EC50 = 500 nM T58921 C6C8NI 44453940 EC50 = 70 nM T58921 C9YUM3 44453941 EC50 = 410 nM T58921 CVI8M4 44453962 EC50 = 130 nM T58921 C63TBK 44453988 EC50 = 30 nM T58921 C5AEL6 44454012 IC50 = 160 nM T58921 C7PA9S 44454244 EC50 = 83 nM T58921 C84FIQ 44454301 EC50 = 50 nM T58921 CIE06L 44454336 EC50 = 2300 nM T58921 CP8OE3 44454364 EC50 = 9400 nM T58921 CA84BK 44454366 EC50 > 10000 nM T58921 CLUF89 44458859 EC50 = 230 nM T58921 CC86GW 44458943 EC50 = 102 nM T58921 CS8EI5 44472992 EC50 = 3800 nM T58921 CR5SI0 44476535 EC50 > 10000 nM T58921 C0ZKT3 44480200 EC50 = 860 nM T58921 C2JMV3 44480201 EC50 = 1400 nM T58921 C42PIO 44480202 EC50 = 13000 nM T58921 CXVI34 44480461 EC50 = 540 nM T58921 C1Y5EX 44480465 EC50 = 5700 nM T58921 CBJ58K 44480717 EC50 = 1500 nM T58921 C89YIZ 44480973 EC50 = 1210 nM T58921 CC1P0L 44481225 EC50 = 1600 nM T58921 CJ6O7D 44481226 EC50 = 3000 nM T58921 CY69AT 44481227 EC50 = 400 nM T58921 C39MBW 44481228 EC50 = 9400 nM T58921 C60RWZ 44481229 EC50 = 720 nM T58921 CEM86S 44481230 EC50 = 870 nM T58921 CO06ZF 44481496 EC50 = 9100 nM T58921 CM4Z1D 44515004 EC50 = 14000 nM T58921 CI4A7H 44515005 IC50 = 2320 nM T58921 CU10OJ 44515008 IC50 = 8100 nM T58921 C75XGY 44543661 EC50 = 53 nM T58921 CU7GD5 44561770 EC50 = 2926 nM T58921 CPW0S4 44561816 EC50 = 27 nM T58921 C9L3VY 44561817 EC50 = 3 nM T58921 C08NKI 44561969 EC50 = 23 nM T58921 CS48WU 44562841 EC50 = 176 nM T58921 C94SYK 44562842 EC50 = 130 nM T58921 CG13BO 44564813 EC50 = 1570 nM T58921 CVN24W 44564853 EC50 = 23 nM T58921 CG1Q3X 44564854 EC50 = 437 nM T58921 CVZA94 44564855 EC50 = 752 nM T58921 CUA0F7 44564899 EC50 = 490 nM T58921 C0VLP9 44564900 EC50 = 7900 nM T58921 C3K9RE 44564901 EC50 = 9270 nM T58921 CBF4N6 44564946 EC50 = 5800 nM T58921 CE16SW 44564947 EC50 = 2190 nM T58921 CEOU52 44565005 EC50 = 560 nM T58921 C9KRL0 44565006 IC50 = 517 nM T58921 C3V0DE 44565017 IC50 = 7140 nM T58921 CB10HQ 44565018 IC50 = 2400 nM T58921 CIY78Z 44565059 IC50 = 7 nM T58921 C12CAF 44565072 IC50 = 12500 nM T58921 C9I2EU 44565119 IC50 = 3400 nM T58921 C4YID3 44565120 IC50 = 3100 nM T58921 C5PN2C 44565121 IC50 = 2390 nM T58921 COW8C0 44565122 IC50 = 33300 nM T58921 CD7P4E 44565166 IC50 = 50000 nM T58921 CCO8N3 44565167 IC50 = 1000000 nM T58921 C0T8MJ 44565168 IC50 = 33300 nM T58921 C1YTC0 44565169 IC50 = 33300 nM T58921 C90ZGD 44571467 EC50 = 560 nM T58921 CC5D2Q 44571468 EC50 = 450 nM T58921 CJ1U6C 44571517 EC50 = 430 nM T58921 CS1M8O 44571518 EC50 = 31 nM T58921 CO5I8F 44571519 EC50 = 100 nM T58921 C9MRZ4 44577533 EC50 = 96 nM T58921 CK32HI 44577534 EC50 = 4096 nM T58921 C7QHB2 44577535 EC50 = 1385 nM T58921 CGF48S 44577684 EC50 = 19.8 nM T58921 C72EIS 44577685 EC50 = 239 nM T58921 CBX3M7 44577687 EC50 = 5010 nM T58921 CSZ15V 44579211 EC50 = 2150 nM T58921 C6NPQ1 44579212 EC50 = 1670 nM T58921 CA9V0O 44579252 EC50 = 5830 nM T58921 CJM4Q7 44579253 EC50 = 1890 nM T58921 CW91PX 44579254 EC50 = 2230 nM T58921 C1E0AL 44579255 EC50 = 7560 nM T58921 CWT1Z0 44579288 EC50 = 3720 nM T58921 CJ82SN 44579289 EC50 = 396 nM T58921 CV2W1S 44579290 EC50 = 2380 nM T58921 C8NIJ4 44579291 EC50 = 3930 nM T58921 C0GH1U 44579338 EC50 = 689 nM T58921 C6S4IV 44579339 EC50 = 174 nM T58921 C1Y4EU 44579340 EC50 = 661 nM T58921 C3JM1U 44579341 EC50 = 706 nM T58921 C4ZX3L 44579390 EC50 = 1440 nM T58921 C45FJV 44579391 EC50 = 670 nM T58921 CE1LR6 44579392 EC50 = 862 nM T58921 CS8N1U 44579393 EC50 = 1420 nM T58921 CU7FR4 44579432 EC50 = 2300 nM T58921 C5A2XS 44579433 EC50 = 3300 nM T58921 C1DJ9V 44579434 EC50 = 12600 nM T58921 C9P4VB 44579435 EC50 = 4600 nM T58921 CLF57W 44579436 EC50 = 2320 nM T58921 C0H9TA 44579477 EC50 = 504 nM T58921 C0KI2H 44579478 EC50 = 728 nM T58921 C10IXM 44579479 EC50 = 5290 nM T58921 C75KTS 44579480 EC50 = 4880 nM T58921 C6R9MQ 44579552 EC50 = 22830 nM T58921 C7LE5D 44579553 EC50 = 18760 nM T58921 C9EB1U 44582932 EC50 = 3 nM T58921 CW72IT 44583199 EC50 = 1 nM T58921 CM8E5G 44584224 Ki = 175.5 nM T58921 CO5RI6 44587736 EC50 = 36 nM T58921 C15RIM 44587737 EC50 = 24 nM T58921 CVI68J 44587738 EC50 = 15 nM T58921 CO3IQ1 44587769 EC50 = 22 nM T58921 CNI3D6 44587770 EC50 = 35 nM T58921 CW67EM 44587801 EC50 = 160 nM T58921 C5JNC0 44589628 EC50 = 15000 nM T58921 C92WZN 44589847 EC50 = 2550 nM T58921 CH5E9L 44589848 EC50 = 2230 nM T58921 CYQ8C5 44589849 EC50 = 2480 nM T58921 CD7ZA0 44589850 EC50 = 8540 nM T58921 CK8L4M 44589851 EC50 = 3680 nM T58921 CUL14S 44589898 EC50 = 4030 nM T58921 C1UQG8 44589954 EC50 = 3160 nM T58921 C35GSR 44589955 EC50 = 2070 nM T58921 CK0A4I 44589956 EC50 = 4360 nM T58921 CAMT56 44589957 EC50 = 1390 nM T58921 CK34ZS 44590001 EC50 = 11300 nM T58921 CH0WD8 44590002 EC50 = 26.92 nM T58921 C2I9QA 44590003 EC50 = 48.98 nM T58921 C4UM8I 44590004 EC50 = 64.57 nM T58921 C8WSC0 44590101 EC50 = 416.87 nM T58921 C5JW0E 44591474 EC50 = 5 nM T58921 CAZD19 44591655 EC50 = 1615 nM T58921 CV3EF4 44591696 EC50 = 716 nM T58921 CI2PD6 44591724 IC50 = 23 nM T58921 COY5U4 44591725 EC50 = 11 nM T58921 CJ6H8E 44591726 EC50 = 10 nM T58921 C68RUE 44591751 EC50 = 21 nM T58921 C08IUA 44591752 EC50 = 4 nM T58921 CBUF12 44591753 IC50 = 3 nM T58921 CJY09Q 44591777 EC50 = 9 nM T58921 C3B5QX 44591778 IC50 = 2 nM T58921 CQH38Y 44591779 IC50 = 3 nM T58921 CQI2P9 44591780 IC50 = 5 nM T58921 CU49SN 44591801 EC50 = 787 nM T58921 CY59XQ 44591802 EC50 = 1210 nM T58921 C0S2NU 44591803 EC50 = 37 nM T58921 CTDI10 44591804 EC50 = 21 nM T58921 CYEN80 44591805 IC50 = 8 nM T58921 C3F5GK 44591814 EC50 = 122 nM T58921 CN3WH7 44591815 EC50 = 33 nM T58921 C7RNC3 44591816 EC50 = 7 nM T58921 CL6FI5 44591830 EC50 = 60 nM T58921 CBX06Y 44601732 EC50 = 73 nM T58921 CH9CK4 44626477 EC50 > 10000 nM T58921 CPW57V 44626478 EC50 > 10000 nM T58921 CUY95T 44626479 EC50 > 10000 nM T58921 CI31DJ 44626480 EC50 > 10000 nM T58921 C8TD4Z 44626481 EC50 > 10000 nM T58921 C0Z3XM 44626583 EC50 > 10000 nM T58921 C3VF6I 44626585 EC50 > 10000 nM T58921 C3ME5P 44626586 EC50 > 10000 nM T58921 CDIP96 44626587 EC50 > 10000 nM T58921 C6V4SD 44626689 EC50 > 10000 nM T58921 CB0GJ9 44626691 EC50 > 10000 nM T58921 CP9YH7 44626696 EC50 > 10000 nM T58921 C01AMG 44626697 EC50 > 10000 nM T58921 CY3I4V 44626789 EC50 > 10000 nM T58921 CXI58P 44626791 EC50 > 10000 nM T58921 C4JRP9 44626797 EC50 > 10000 nM T58921 C3YK1M 44626798 EC50 > 10000 nM T58921 C3Q2XF 44626799 EC50 > 10000 nM T58921 CB1ZX0 44626800 EC50 > 10000 nM T58921 C4A0WS 44626801 EC50 > 10000 nM T58921 C6EF1Q 44626888 EC50 > 10000 nM T58921 C6X8KS 44626889 EC50 > 10000 nM T58921 C5I8NM 44626890 EC50 > 10000 nM T58921 C8V9SP 44626891 EC50 > 10000 nM T58921 CTY31Z 44626892 EC50 > 10000 nM T58921 CQI69K 44626986 EC50 > 10000 nM T58921 C8NAD5 44626987 EC50 > 10000 nM T58921 C0RAL3 44626988 EC50 > 10000 nM T58921 C4BNA9 44626989 EC50 > 10000 nM T58921 CQ5O3I 44626990 EC50 > 10000 nM T58921 CESB05 44627078 EC50 = 5660 nM T58921 CSW84C 44627079 EC50 = 6890 nM T58921 C3ZM7B 44627080 EC50 = 6360 nM T58921 C6B2RO 44627083 EC50 > 10000 nM T58921 C2JB5Y 44627084 EC50 > 10000 nM T58921 CABC27 44627085 EC50 > 10000 nM T58921 CPS63M 44627086 EC50 = 1200 nM T58921 CX41JP 44627087 EC50 = 1560 nM T58921 CL34OS 44627188 EC50 > 10000 nM T58921 CCQ59P 44627190 EC50 > 10000 nM T58921 CMG9Q4 44627191 EC50 > 10000 nM T58921 C9OI6W 44627192 EC50 > 10000 nM T58921 CQJ26Z 44627297 EC50 > 10000 nM T58921 C87MHR 44627298 EC50 > 10000 nM T58921 C5W3IT 44627299 EC50 > 10000 nM T58921 CS25FR 44627300 EC50 > 10000 nM T58921 C0SYJ8 44627301 EC50 > 10000 nM T58921 CY49NK 44627302 EC50 > 10000 nM T58921 C6RBQ1 44627303 EC50 > 10000 nM T58921 CUL63M 44627304 EC50 > 10000 nM T58921 C1G2QK 44627305 EC50 > 10000 nM T58921 C96QCO 44627306 EC50 > 10000 nM T58921 CR8A1I 44627407 EC50 > 10000 nM T58921 CE2J5V 44627408 EC50 > 10000 nM T58921 C43ZOX 44627409 EC50 > 10000 nM T58921 C7K0GI 44627410 EC50 > 10000 nM T58921 CA31WU 44627411 EC50 > 10000 nM T58921 CPY46S 44627412 EC50 > 10000 nM T58921 CI1VN2 44627413 EC50 > 10000 nM T58921 CK83HR 44627414 EC50 > 10000 nM T58921 C1DQ7N 44627415 EC50 > 10000 nM T58921 CF1Q5E 44627416 EC50 > 10000 nM T58921 CPFN63 44627417 EC50 = 2490 nM T58921 C9TNL0 44627524 EC50 > 10000 nM T58921 C3OXU2 44627525 EC50 > 10000 nM T58921 C3PZ6T 44627526 EC50 > 10000 nM T58921 CD47HB 44627527 EC50 > 10000 nM T58921 C1KAJ2 44627528 EC50 > 10000 nM T58921 CR93CX 44627529 EC50 = 1030 nM T58921 CY95DP 44627531 EC50 > 10000 nM T58921 CD8L4U 44627532 EC50 > 10000 nM T58921 CYJ52X 44627533 EC50 > 10000 nM T58921 CJ43OZ 44627627 EC50 > 10000 nM T58921 CEA3I2 44627628 EC50 > 10000 nM T58921 CW7PG6 44627633 EC50 > 10000 nM T58921 CX0Q2Y 44627634 EC50 = 1310 nM T58921 CIWZ13 44627635 EC50 > 10000 nM T58921 CA4W0L 44627636 EC50 > 10000 nM T58921 C28SEU 44627637 EC50 > 10000 nM T58921 C6D0XF 44627728 EC50 > 10000 nM T58921 CAQ41R 44627729 EC50 > 10000 nM T58921 CCN8S2 44627730 EC50 > 10000 nM T58921 CGO41A 44627731 EC50 > 10000 nM T58921 C1HMU7 44627732 EC50 > 10000 nM T58921 C8K3GF 44627733 EC50 > 10000 nM T58921 C3T1HB 44627734 EC50 > 10000 nM T58921 CE93BG 44627735 EC50 > 10000 nM T58921 CPFV72 44627838 EC50 > 10000 nM T58921 CEH41N 44627839 EC50 > 10000 nM T58921 C2SJ5A 44627840 EC50 > 10000 nM T58921 C53AJB 44627841 EC50 > 10000 nM T58921 CXHP05 44627842 EC50 > 10000 nM T58921 CZL75R 44627843 EC50 > 10000 nM T58921 CRI4Q6 44627844 EC50 > 10000 nM T58921 CK7Z9X 44627845 EC50 > 10000 nM T58921 C95MPI 44627846 EC50 > 10000 nM T58921 C8SPR5 44627847 EC50 > 10000 nM T58921 C2LI9T 44627941 EC50 > 10000 nM T58921 CA8CB6 44627942 EC50 > 10000 nM T58921 CSDF01 44627943 EC50 > 10000 nM T58921 CM5D8L 44627944 EC50 > 10000 nM T58921 CX23ZO 44627945 EC50 > 10000 nM T58921 C35WJV 44627946 EC50 > 10000 nM T58921 CP9G7C 44627948 EC50 = 600 nM T58921 C6JXF9 44628046 EC50 > 10000 nM T58921 CQX2E8 44628047 EC50 > 10000 nM T58921 CW2I4H 44628048 EC50 > 10000 nM T58921 CUHD90 44628049 EC50 > 10000 nM T58921 C24MHW 44628050 EC50 > 10000 nM T58921 CG3B8F 45102750 EC50 = 212 nM T58921 CI7SM1 45104339 IC50 > 10000 nM T58921 C0OX9J 45104340 IC50 > 10000 nM T58921 CB7ED5 45104341 IC50 > 10000 nM T58921 CLFU74 45104342 IC50 > 10000 nM T58921 COD76Z 45104343 IC50 > 10000 nM T58921 CGB9R5 45104439 IC50 > 10000 nM T58921 CNEV35 45104440 IC50 > 10000 nM T58921 CP7L6H 45104441 IC50 > 10000 nM T58921 CF1Y2V 45104442 IC50 > 10000 nM T58921 C8L5CG 45104443 IC50 > 10000 nM T58921 CRIS28 45104444 IC50 > 10000 nM T58921 CTWC94 45104445 IC50 > 10000 nM T58921 C0AHF2 45107476 EC50 = 10400 nM T58921 C4KRT0 45254002 EC50 = 963 nM T58921 CVL46G 45263732 IC50 = 1410 nM T58921 CSLZ04 45267718 EC50 = 3000 nM T58921 C0R8MQ 45267726 EC50 = 4100 nM T58921 CK31XL 45268054 EC50 = 7 nM T58921 CC7X2D 45268061 Ki > 10000 nM T58921 C4A7GC 45268062 Ki = 33 nM T58921 C8AXK3 45268597 EC50 = 4600 nM T58921 C0F7RJ 45268611 EC50 = 4200 nM T58921 C1EIF5 45269442 EC50 = 1600 nM T58921 CU91HN 45269452 EC50 = 540 nM T58921 C74OGR 45269453 EC50 = 15700 nM T58921 CS7EC0 45269787 EC50 = 7.52 nM T58921 CTOB26 45270070 EC50 = 5540 nM T58921 C4X8NT 45270286 EC50 = 5300 nM T58921 CJC3M7 45270291 EC50 = 1300 nM T58921 CTX61C 45271105 EC50 = 9900 nM T58921 C5U8HX 45271112 EC50 = 7800 nM T58921 CZU9Q3 45271445 EC50 = 14 nM T58921 C3PD0Q 45271739 EC50 >= 50000 nM T58921 CR1QU8 45271974 EC50 = 2600 nM T58921 CN4ET7 45271983 EC50 = 2300 nM T58921 CH92UP 45271992 EC50 = 1200 nM T58921 CNU0H3 45272171 IC50 = 1 nM T58921 CTFJ48 45272617 EC50 = 5010 nM T58921 C42QTW 45272810 EC50 = 930 nM T58921 CVU12R 45272820 EC50 = 8100 nM T58921 CXS0Y5 45273207 EC50 = 13 nM T58921 CYN5B1 45273613 EC50 >= 50000 nM T58921 COP75F 45273770 EC50 = 3000 nM T58921 CQ4GE9 45273780 EC50 = 3800 nM T58921 CM3Q4K 45482771 EC50 = 2400 nM T58921 CO1GI5 45482833 EC50 = 870 nM T58921 C72CNH 45783216 Ki = 700 nM T58921 C89QTJ 46184983 EC50 = 292 nM T58921 CFA6V5 46196683 EC50 = 843 nM T58921 C9JV0C 46196684 EC50 = 1482 nM T58921 CB4MV0 46196685 EC50 = 905 nM T58921 CJG9N2 46196686 EC50 = 826 nM T58921 C9ZV8D 46196687 EC50 = 1257 nM T58921 C1GER0 46197994 EC50 = 75.4 nM T58921 CMJ12Z 46197995 EC50 = 41.5 nM T58921 CEGI58 46197996 EC50 = 141.2 nM T58921 CYAI40 46198106 EC50 = 2901 nM T58921 CTI0F8 46198107 EC50 = 1411 nM T58921 CJ9OY8 46198108 EC50 = 2500 nM T58921 CI9QH8 46198109 EC50 = 1100 nM T58921 CU3VQ1 46198110 IC50 = 384 nM T58921 C2P9ST 46198216 EC50 = 1007 nM T58921 C3NFH5 46198217 EC50 = 20.1 nM T58921 CWR39G 46198218 EC50 = 398 nM T58921 CV8B3T 46198219 EC50 = 417 nM T58921 CSEL57 46198325 EC50 = 3445 nM T58921 C2VIF3 46198326 EC50 = 1124 nM T58921 C6JWH5 46198327 EC50 = 684 nM T58921 CIJN79 46198328 EC50 = 284 nM T58921 C13RUW 46198329 EC50 = 705 nM T58921 CY97NP 46213107 EC50 = 21 nM T58921 C5D9KI 46216831 EC50 = 1100 nM T58921 CS4K6Y 46216832 EC50 = 1600 nM T58921 CSR2C5 46226840 Ki = 1.83 nM T58921 C01JNB 46226841 Ki = 0.17 nM T58921 CF80GU 46228280 IC50 = 18000 nM T58921 C5E2FZ 46228281 IC50 = 14000 nM T58921 C0ZWT3 46229787 EC50 = 1400 nM T58921 C2VBA4 46229788 EC50 = 2100 nM T58921 CT9JR4 46229789 EC50 = 1400 nM T58921 COI07L 46229832 EC50 = 1900 nM T58921 C7M2LT 46229833 EC50 = 200 nM T58921 C2C4EF 46229834 EC50 = 100 nM T58921 C2OCX1 46229835 EC50 = 200 nM T58921 C3DY0A 46229869 EC50 = 200 nM T58921 CFTW35 46229870 EC50 = 800 nM T58921 CNE12J 46229871 EC50 = 1000 nM T58921 C1O2HJ 46229903 EC50 = 700 nM T58921 C2R8WH 46232959 EC50 = 900 nM T58921 C12JOZ 46232960 EC50 = 163 nM T58921 CL36PQ 46233001 EC50 = 17 nM T58921 C3Q6DN 46233002 EC50 = 0.8 nM T58921 C0P5ED 46233003 IC50 = 1 nM T58921 C19XSC 46233038 IC50 = 18 nM T58921 CBSA69 46233039 EC50 = 1 nM T58921 C5O7FJ 46233040 EC50 = 338 nM T58921 CE93XQ 46233070 EC50 = 2 nM T58921 C9A2QS 46233071 EC50 = 3 nM T58921 CT53DY 46233072 EC50 = 201 nM T58921 C2RTO6 46837638 EC50 = 6100 nM T58921 CM2K0V 46837639 EC50 = 8800 nM T58921 C2OP7F 46837642 EC50 = 8900 nM T58921 CHJD18 46837643 EC50 = 10000 nM T58921 CIH0K4 46837775 EC50 = 7500 nM T58921 CV5ZO3 46837777 EC50 = 11000 nM T58921 CWFQ46 46837778 EC50 = 10300 nM T58921 CEPL58 46837915 EC50 = 7000 nM T58921 CM3H5J 46837918 EC50 = 6600 nM T58921 CKDW89 46837919 EC50 = 12100 nM T58921 CD5UE3 46837920 EC50 = 4300 nM T58921 C4S6ID 46838058 EC50 = 11000 nM T58921 CQXV17 46838061 EC50 = 10400 nM T58921 CR9M7C 46845962 Ki = 43000 nM T58921 C6YQ7W 46845963 Ki = 43600 nM T58921 CB5IQ7 46845964 Ki = 7300 nM T58921 CD1W9S 46845965 Ki = 4000 nM T58921 C6C0JN 46846227 IC50 = 2 nM T58921 CT9HY5 46854103 EC50 = 180 nM T58921 C6FL4H 46854264 EC50 = 1600 nM T58921 CYPW28 46854265 EC50 = 670 nM T58921 C2X3YD 46854432 EC50 = 250 nM T58921 C0K8XB 46854433 EC50 = 740 nM T58921 C50WIR 46854434 EC50 = 2700 nM T58921 CZ1CF5 46854435 EC50 > 10000 nM T58921 CZ2S8I 46854436 EC50 > 10000 nM T58921 CV50PY 46854437 EC50 = 1800 nM T58921 CG2H0F 46854438 EC50 = 300 nM T58921 C1GM0O 46854597 EC50 > 10000 nM T58921 CIK92N 46854598 EC50 = 2300 nM T58921 CYXR46 46854599 EC50 = 470 nM T58921 CMZ6H4 46854600 EC50 = 250 nM T58921 CZTG82 46854601 EC50 = 420 nM T58921 COW60Q 46854602 EC50 > 10000 nM T58921 CXYW03 46854747 EC50 > 10000 nM T58921 CVZ97H 46861800 EC50 = 772 nM T58921 C57NTP 46866189 EC50 = 4500 nM T58921 CET7R4 46866190 EC50 = 7800 nM T58921 CE72MC 46878644 EC50 > 10000 nM T58921 C4WDX1 46878645 EC50 = 2300 nM T58921 C1QT8Z 46878727 EC50 = 2560 nM T58921 CWZ8N4 46878728 EC50 = 4610 nM T58921 C4WO1G 46878729 EC50 = 5870 nM T58921 CRK26D 46878777 EC50 > 10000 nM T58921 C0HYG2 46878778 EC50 > 10000 nM T58921 C49SRK 46878779 EC50 > 10000 nM T58921 C62JTF 46878780 EC50 > 10000 nM T58921 C3OZP9 46878781 EC50 > 10000 nM T58921 C51RAC 46878843 EC50 > 10000 nM T58921 CDL01S 46880009 IC50 = 10 nM T58921 CG3D5X 46880447 EC50 > 100000 nM T58921 CD05FS 46884868 EC50 = 50220 nM T58921 C08GUA 46885478 EC50 = 6900 nM T58921 CB6X5P 46885522 EC50 = 7600 nM T58921 CL92SR 46885552 EC50 = 7300 nM T58921 CSU0B6 46885553 EC50 = 9000 nM T58921 CC14YP 46885554 EC50 = 13000 nM T58921 CA78QN 46885556 EC50 = 8900 nM T58921 CPI5N2 46885589 EC50 = 10800 nM T58921 CP3EV2 46885590 EC50 = 8900 nM T58921 C7C6LI 46885591 EC50 = 6800 nM T58921 CF65OR 46888895 EC50 = 9193 nM T58921 C0S8WL 46888896 EC50 = 4815 nM T58921 CB3FC1 46888897 EC50 = 15580 nM T58921 C5MH4J 46888966 EC50 > 25000 nM T58921 CIQT59 46888967 EC50 > 25000 nM T58921 CRJ67A 46888968 EC50 > 25000 nM T58921 C20VWR 46888969 EC50 > 25000 nM T58921 CGI9Q8 46888992 EC50 = 6386 nM T58921 C3ZG7B 46888993 EC50 > 8300 nM T58921 C2MO0J 46888994 EC50 = 20690 nM T58921 CJB37Y 46888995 EC50 = 4692 nM T58921 C4N7ZM 46889020 EC50 = 9288 nM T58921 CV0O3M 46889021 EC50 > 25000 nM T58921 C0IVK1 46889022 EC50 = 4018 nM T58921 CCNZ52 46889045 EC50 = 5036 nM T58921 CZ1H2N 46889046 EC50 = 1692 nM T58921 CU9R0D 46889047 EC50 = 571 nM T58921 C6TQX2 46889072 EC50 = 970 nM T58921 CJ3V7K 46889073 EC50 = 710 nM T58921 CQJ70A 46889074 EC50 = 1444 nM T58921 C0H6FU 46908722 EC50 = 200 nM T58921 CL0R6B 46908814 EC50 = 176 nM T58921 C4FAD6 46908815 EC50 = 24 nM T58921 CI7U3G 46908816 EC50 = 21 nM T58921 C2QIR9 46908817 EC50 = 89 nM T58921 CRF0E4 46908818 EC50 = 100 nM T58921 C6VB0S 46908904 EC50 = 43 nM T58921 C3NMP1 46908905 EC50 = 41 nM T58921 CMV76P 46911693 EC50 = 1720 nM T58921 C86WTO 46911745 EC50 = 172 nM T58921 CN9L7G 46916268 EC50 > 15000 nM T58921 CS13YQ 49846481 IC50 > 100000 nM T58921 CUD91T 49862248 EC50 = 1450000 nM T58921 C7ZBL0 49863999 EC50 = 400 nM T58921 C2MDF4 49864012 EC50 = 470 nM T58921 C2Q1UG 49864013 EC50 = 400 nM T58921 CE25VJ 49864014 EC50 = 580 nM T58921 CO0H5D 49864015 EC50 = 620 nM T58921 CA5WO8 49864025 EC50 = 2900 nM T58921 C8XHF0 49864026 EC50 = 3500 nM T58921 CMV2E1 49910818 EC50 = 11000 nM T58921 C0Z6EF 49913435 EC50 = 10000 nM T58921 CSBV96 50898774 EC50 = 340 nM T58921 C8MF9U 50925432 EC50 = 3.6 nM T58921 CP3Y0J 50925503 EC50 > 1000 nM T58921 CD2G5X 50925504 EC50 = 290.3 nM T58921 C4PK6S 50942697 EC50 > 20000 nM T58921 C96HOP 50942698 EC50 = 800 nM T58921 CZHE17 50994601 EC50 = 3.6 nM T58921 CK03LY 51038993 EC50 = 1700 nM T58921 CT59YM 51039006 EC50 = 500 nM T58921 CZ23XJ 51049637 IC50 = 24 nM T58921 CNVB53 51346913 EC50 = 800 nM T58921 CAXJ10 52918120 IC50 = 6309.57 nM T58921 CRN19G 52918121 IC50 = 6309.57 nM T58921 C3TJ7N 52921716 IC50 = 7 nM T58921 C3KM6T 53233135 EC50 = 0.018 nM T58921 C7AJ1Q 53239853 EC50 = 516 nM T58921 CK3RV4 53239854 IC50 = 80 nM T58921 CKD21Q 53239857 IC50 = 4 nM T58921 CN8H7B 53240432 EC50 = 130 nM T58921 CJX25Z 53249102 EC50 = 220000 nM T58921 C6F2KY 53309128 EC50 = 175 nM T58921 C9SA4X 53309129 EC50 = 1320 nM T58921 C07WMK 53309130 EC50 = 295 nM T58921 CLV60X 53309271 EC50 = 762 nM T58921 C0SL6H 53309272 EC50 = 1820 nM T58921 CBPQ05 53309273 EC50 = 1340 nM T58921 CR3N6U 53309274 EC50 = 494 nM T58921 CA97CK 53309275 EC50 = 264 nM T58921 CI6KE2 53309404 EC50 = 89 nM T58921 C1EM8J 53309405 EC50 = 165 nM T58921 C0EH4S 53309406 EC50 = 90 nM T58921 CL83BY 53317593 EC50 = 270.6 nM T58921 CVN51I 53317892 EC50 = 100.2 nM T58921 CTUA27 53317893 EC50 > 1000 nM T58921 C4H5CJ 53319204 EC50 = 2000 nM T58921 C7I9UO 53319246 EC50 > 1000 nM T58921 C1JIB3 53319416 EC50 > 30000 nM T58921 C8JL7M 53323370 EC50 = 2700 nM T58921 C3PYV7 53325836 EC50 > 1000 nM T58921 CDS84F 53362000 EC50 = 852 nM T58921 C9DJI4 53362018 EC50 = 1141 nM T58921 CC7KT6 53363130 EC50 = 3400 nM T58921 CF5U2R 53363131 EC50 = 4800 nM T58921 CSC3V7 53363132 EC50 = 4700 nM T58921 CH2DO7 53363133 EC50 = 7800 nM T58921 CPD82G 53363134 EC50 = 3700 nM T58921 CI4D2P 53363220 EC50 = 2200 nM T58921 CX7I2Y 53363222 EC50 = 10800 nM T58921 C1WB4D 53363224 EC50 = 1800 nM T58921 CUI04W 53363313 EC50 = 7200 nM T58921 CK5IH6 53389233 IC50 = 3 nM T58921 CU7D6G 53389234 EC50 = 116 nM T58921 C56PQL 53389239 EC50 = 185 nM T58921 CT8A1D 53389242 IC50 = 5 nM T58921 CYM6X2 53389244 EC50 = 133 nM T58921 C25IBL 53389250 EC50 = 355 nM T58921 CA82BQ 53389252 EC50 = 226 nM T58921 C02RVT 53481926 EC50 = 100 nM T58921 CE86AX 53481931 IC50 = 5 nM T58921 CV9W4N 53481932 EC50 = 344 nM T58921 CJ0DI2 53481933 IC50 = 97 nM T58921 C0EM7R 54178446 EC50 = 591 nM T58921 CAKC25 54579783 IC50 = 8 nM T58921 C93CGK 54579786 Ki = 32225 nM T58921 CL2VM8 54579977 IC50 = 3981.07 nM T58921 CV9U5K 54580014 IC50 = 6309.57 nM T58921 C9IN5X 54580015 IC50 = 3162.28 nM T58921 C64SWC 54580016 IC50 = 5011.87 nM T58921 COD82I 54580272 IC50 = 56 nM T58921 CN0U2D 54580274 IC50 = 540 nM T58921 C2HE7A 54580445 EC50 = 620000000 nM T58921 C76WZO 54580529 EC50 = 780 nM T58921 C6M9HP 54580530 EC50 = 830 nM T58921 CKBG47 54580531 EC50 = 990 nM T58921 CSH41U 54580814 EC50 = 5900 nM T58921 C8MLC0 54580964 IC50 = 2511.89 nM T58921 C8EUF2 54580965 IC50 = 3162.28 nM T58921 CM6I8P 54580966 IC50 = 6309.57 nM T58921 CR5DC6 54580967 IC50 = 6309.57 nM T58921 CPT96V 54581011 IC50 = 3981.07 nM T58921 C2E5NY 54581038 EC50 = 4600 nM T58921 CM95BU 54581270 IC50 = 76 nM T58921 CSU6T3 54581271 IC50 = 490 nM T58921 CO40YF 54581272 IC50 = 450 nM T58921 CV82WR 54581273 IC50 = 640 nM T58921 CH0Z2K 54581274 IC50 = 1760 nM T58921 CDP3R7 54581456 EC50 = 40000000 nM T58921 C81THX 54581535 EC50 = 920 nM T58921 CBE79V 54581857 EC50 = 31100 nM T58921 CAT03Y 54582018 IC50 = 7943.28 nM T58921 CMLX87 54582047 IC50 = 6309.57 nM T58921 CV2YZ7 54582292 IC50 = 195 nM T58921 CY0DS9 54582293 IC50 = 46 nM T58921 COK58J 54582294 IC50 = 750 nM T58921 CRKL15 54582795 EC50 = 26400 nM T58921 CT4IJ9 54582796 EC50 = 5100 nM T58921 CQ89ZY 54582993 IC50 = 7943.28 nM T58921 CP92OU 54582994 IC50 = 10000 nM T58921 CGTN92 54582995 IC50 = 5011.87 nM T58921 C18HFY 54583023 EC50 = 6000 nM T58921 C9RSW3 54583265 IC50 = 30 nM T58921 CH2QL0 54583266 IC50 = 735 nM T58921 CCH3I6 54583267 IC50 = 1160 nM T58921 C41XBG 54583268 IC50 = 57 nM T58921 CHQ79P 54583754 EC50 = 25100 nM T58921 C1D5YV 54583795 EC50 = 19100 nM T58921 CK48SJ 54583995 IC50 = 3981.07 nM T58921 C9YDX0 54583996 IC50 = 7943.28 nM T58921 CX1V3U 54583997 IC50 = 5011.87 nM T58921 CGXM65 54583998 IC50 = 7943.28 nM T58921 CS36HY 54584012 IC50 = 144 nM T58921 CJH31Y 54584032 EC50 = 3300 nM T58921 C7YX6S 54584227 IC50 = 37 nM T58921 C94QXU 54584228 IC50 = 85 nM T58921 CPA4F6 54584229 IC50 = 63 nM T58921 C9JSC0 54584230 IC50 = 170 nM T58921 C1M6EB 54584231 IC50 = 77 nM T58921 CX2D0T 54584232 IC50 = 1845 nM T58921 CBP42C 54584463 Ki = 118850222.7 nM T58921 CK6CI7 54584935 IC50 = 6309.57 nM T58921 C1KOF7 54584936 IC50 = 3981.07 nM T58921 CPXG09 54584937 IC50 = 5011.87 nM T58921 CBO34V 54584938 IC50 = 1584.89 nM T58921 C02CRJ 54584979 EC50 > 10000 nM T58921 C7PD4R 54585193 IC50 = 291 nM T58921 CD51LU 54585194 IC50 = 59 nM T58921 C2AI3Y 54585195 IC50 = 73 nM T58921 C82UFZ 54585196 IC50 = 78 nM T58921 CGE26L 54585197 IC50 = 6440 nM T58921 CNO4C1 54585198 IC50 = 1845 nM T58921 CH9M7S 54585199 IC50 = 180 nM T58921 CQU27M 54585710 EC50 > 10000 nM T58921 C4DX7E 54585711 EC50 = 2600 nM T58921 C3TU7R 54585867 IC50 = 7943.28 nM T58921 COX28A 54585896 IC50 = 6309.57 nM T58921 C6ZSM0 54585897 IC50 = 5011.87 nM T58921 CXL71T 54585898 IC50 = 3162.28 nM T58921 C7D1LE 54585899 IC50 = 5011.87 nM T58921 C0I2DH 54585900 IC50 = 12589.25 nM T58921 CP8F9I 54585901 IC50 = 7943.28 nM T58921 C0JOG1 54585902 IC50 = 1995.26 nM T58921 C9Q0VG 54585903 IC50 = 5011.87 nM T58921 CU43ME 54585904 IC50 = 6309.57 nM T58921 CFZ6E9 54585935 EC50 = 12000 nM T58921 CO0XN5 54585936 EC50 = 1700 nM T58921 CRUV25 54586152 IC50 = 1087 nM T58921 C3VMX8 54586154 IC50 = 300 nM T58921 CW0L9M 54586395 EC50 > 10000 nM T58921 C6EC0W 54586396 EC50 = 460 nM T58921 CO0X2A 54586658 EC50 = 20800 nM T58921 CM9GL4 54586691 EC50 > 10000 nM T58921 C8NZ6D 54586832 IC50 = 5011.87 nM T58921 C18JYB 54586833 IC50 = 5011.87 nM T58921 C2K6FY 54586870 IC50 = 5011.87 nM T58921 C8UO7K 54586871 IC50 = 7943.28 nM T58921 CTL0F5 54586872 IC50 = 6309.57 nM T58921 C28UYH 54586873 IC50 = 5011.87 nM T58921 CF3BK8 54586906 EC50 = 4800 nM T58921 CP6D9X 54586907 EC50 = 3000 nM T58921 CM92IS 54587159 IC50 = 335 nM T58921 C7XD2U 54587160 IC50 = 226 nM T58921 CQV09E 54587161 IC50 = 30 nM T58921 C1QY8H 54587162 IC50 = 1851 nM T58921 C7N0YU 54587410 EC50 = 4600 nM T58921 C14QDZ 54587728 EC50 > 10000 nM T58921 C5J0BW 54587729 EC50 = 1000 nM T58921 C5ZX4B 54597874 IC50 > 10000 nM T58921 CRN5D3 54764927 EC50 > 1000 nM T58921 C8B9NI 56658065 EC50 = 398.11 nM T58921 CKIC64 56659331 EC50 = 8500 nM T58921 CRB95Z 56659332 EC50 = 7900 nM T58921 C92XSL 56659333 EC50 = 6900 nM T58921 CT1A3Y 56659334 EC50 = 5200 nM T58921 CA9U3S 56659347 EC50 = 0.0015 nM T58921 CF29WQ 56659348 EC50 = 0.0002 nM T58921 C0N9SG 56661577 EC50 = 10000 nM T58921 CMK23G 56665220 EC50 = 1500 nM T58921 C4CP6U 56666265 EC50 = 11000 nM T58921 CIUN54 56666266 EC50 = 7100 nM T58921 C7NA3W 56666267 EC50 = 3200 nM T58921 C7IW4Z 56669680 EC50 = 12000 nM T58921 CGP42W 56669681 EC50 = 9300 nM T58921 C5I0GB 56669682 EC50 = 6900 nM T58921 C1MAL6 56669688 EC50 = 2.7 nM T58921 CVQ64B 56669689 EC50 = 0.05 nM T58921 C50PUC 56669690 EC50 = 0.0001 nM T58921 CAM0T3 56671941 EC50 = 5011.87 nM T58921 C8M1KV 56671942 EC50 = 398.11 nM T58921 CP1ES6 56672150 EC50 = 1100 nM T58921 CN8YH0 56673196 EC50 = 4.5 nM T58921 C8E7PL 56675543 EC50 = 2500 nM T58921 CQ58IX 56676515 EC50 = 17000 nM T58921 CV6Z3S 56676516 EC50 = 12000 nM T58921 C1H5IV 56676523 EC50 = 3 nM T58921 CV12UQ 56679849 EC50 = 0.0003 nM T58921 CKLC32 56679850 EC50 = 0.6 nM T58921 CXMR78 56925781 EC50 = 3000 nM T58921 C5HQZ6 56925892 EC50 = 489 nM T58921 C0NRU5 56925893 EC50 = 135 nM T58921 C2B6MF 56925894 IC50 = 1374 nM T58921 CJ46YQ 56925895 EC50 = 200 nM T58921 CR6TP4 56925896 EC50 = 4.1 nM T58921 CVO3A2 56925994 EC50 = 3000 nM T58921 CLCM62 56925995 EC50 = 77.5 nM T58921 C8GLC1 56925996 IC50 = 35.4 nM T58921 C2M8DR 56925997 IC50 = 4.1 nM T58921 CD75ZU 56925998 IC50 = 3.2 nM T58921 C8YGX7 56926094 IC50 = 2.3 nM T58921 C15OKZ 56926095 IC50 = 4.1 nM T58921 CN68DG 56926096 IC50 = 66 nM T58921 C4K1XH 56926097 EC50 = 102 nM T58921 CFO3R4 56926098 IC50 = 924 nM T58921 C7X3WK 56926185 IC50 = 3657 nM T58921 CZEF98 56926186 IC50 = 6633 nM T58921 C92DPX 56926187 IC50 = 2177 nM T58921 CSJW15 56926188 IC50 = 6935 nM T58921 C9VTF3 56926189 EC50 = 2 nM T58921 CMK92V 56926276 EC50 = 8 nM T58921 COT54N 56929220 EC50 = 9.2 nM T58921 COP96Y 56929315 EC50 = 34 nM T58921 CG4H5R 56929316 EC50 = 12 nM T58921 C7TI8R 56929317 EC50 = 22 nM T58921 CC59QX 56929500 EC50 = 34.6 nM T58921 C51UMZ 56929501 EC50 = 65.2 nM T58921 C1RFK2 56929502 EC50 = 52.7 nM T58921 C05HRD 56929503 EC50 = 49.5 nM T58921 C3H9GM 56929596 EC50 = 28.7 nM T58921 C7F2WU 56929598 EC50 = 73.8 nM T58921 CDY7W8 56929599 EC50 = 85.9 nM T58921 CNB56J 56940812 EC50 > 10000 nM T58921 CA7Y1Z 56941393 EC50 > 10000 nM T58921 C1DQ4M 56942395 EC50 > 10000 nM T58921 CN5Z9T 56945389 EC50 = 150 nM T58921 CNC6B5 56945390 EC50 = 800 nM T58921 CI6L5H 56945391 EC50 = 2700 nM T58921 CRJC63 56945487 EC50 = 2300 nM T58921 CPSB16 56945488 EC50 = 1700 nM T58921 C0MC8V 56949691 EC50 = 12 nM T58921 CQ19IH 56949692 EC50 = 9.3 nM T58921 CB4F9K 56949693 EC50 = 8.3 nM T58921 C93NTK 57345550 EC50 = 1880 nM T58921 CWQY91 57345616 EC50 = 500 nM T58921 CP89DR 57390390 EC50 = 2400 nM T58921 CCK42T 57390448 EC50 = 35200 nM T58921 C6SJH9 57390449 EC50 = 14100 nM T58921 C9SB5K 57390812 EC50 > 19000 nM T58921 CIFN56 57391546 EC50 = 10 nM T58921 C8Y0ET 57391547 EC50 = 13 nM T58921 CN5A1Q 57391733 EC50 = 40 nM T58921 CW90NK 57391788 EC50 = 760 nM T58921 CA8SE6 57392192 EC50 = 11600 nM T58921 C96EIM 57392586 EC50 > 13000 nM T58921 CT3U5R 57392587 EC50 > 9800 nM T58921 CIVL69 57392628 EC50 > 12000 nM T58921 CX8QN1 57392629 EC50 > 6800 nM T58921 C7A2XY 57392630 EC50 > 9800 nM T58921 C5JD9O 57392836 EC50 = 5900 nM T58921 CLDQ51 57393295 EC50 = 16 nM T58921 C5I1CA 57393296 EC50 = 150 nM T58921 C5A7HW 57393297 EC50 = 31 nM T58921 CR3Y5U 57393471 EC50 = 240 nM T58921 C9OCN0 57393518 EC50 = 760 nM T58921 CB01SO 57393940 EC50 = 32000 nM T58921 C5BG1A 57394147 EC50 > 1000 nM T58921 CK5HD6 57394349 EC50 > 10000 nM T58921 CZ0Y1N 57394350 EC50 > 6800 nM T58921 CX34SN 57394351 EC50 > 13000 nM T58921 CV5C3D 57395027 EC50 = 500 nM T58921 C7Q3IB 57395028 EC50 = 110 nM T58921 CE6W5J 57395192 EC50 = 30 nM T58921 CL3O6H 57395194 EC50 = 20 nM T58921 CT45EM 57395675 EC50 = 4900 nM T58921 CHM9Q5 57395750 EC50 = 19000 nM T58921 CHRX78 57396101 EC50 = 3100 nM T58921 C9V1KC 57396779 EC50 = 21 nM T58921 CQ71JU 57396780 EC50 = 17 nM T58921 C8HO1P 57396781 EC50 = 260 nM T58921 CLI70F 57396782 EC50 = 9 nM T58921 C7YC4Z 57396783 EC50 = 8.2 nM T58921 CQJ01F 57396784 EC50 = 160 nM T58921 C56JAF 57396972 EC50 = 50 nM T58921 C6WY1Q 57396974 EC50 = 20 nM T58921 CHEM09 57396976 EC50 = 50 nM T58921 C1D7YR 57397473 EC50 = 16400 nM T58921 C5ZCT7 57397527 EC50 = 41000 nM T58921 C1YTG9 57397528 EC50 = 30000 nM T58921 C2DOZ9 57397718 EC50 > 1000 nM T58921 C3O8JG 57398546 EC50 = 14 nM T58921 C6ET7R 57398547 EC50 = 8.4 nM T58921 C1DPW9 57398548 EC50 = 13 nM T58921 C19KAD 57398549 EC50 = 11 nM T58921 CKL3A8 57398721 EC50 = 30 nM T58921 C9VOI8 57398723 EC50 = 40 nM T58921 CT1GD4 57398727 EC50 = 90 nM T58921 C1DG8N 57398729 EC50 = 70 nM T58921 C3Q9DA 57398755 EC50 = 70 nM T58921 C8HB5R 57399155 EC50 = 5800 nM T58921 CKYR74 57399206 EC50 = 15900 nM T58921 CPX5Z8 57399207 EC50 = 2500 nM T58921 CU6LA3 57399208 EC50 = 900 nM T58921 CPV28C 57399559 EC50 > 15000 nM T58921 CQT4G5 57400212 EC50 = 40 nM T58921 CQC7F9 57400214 EC50 = 120 nM T58921 C8YL6R 57400215 EC50 = 450 nM T58921 C9G7RH 57400394 EC50 = 110 nM T58921 CH0Y4N 57400437 EC50 = 350 nM T58921 CF8QD0 57400441 EC50 = 20 nM T58921 CH5AK1 57400966 EC50 = 3500 nM T58921 CVXB34 57400967 EC50 = 5200 nM T58921 CXO3V1 57401284 EC50 > 13000 nM T58921 C82NSD 57401312 EC50 > 11000 nM T58921 CN1UC5 57402016 EC50 = 29 nM T58921 CTWX97 57402017 EC50 = 20 nM T58921 CY27OL 57402190 EC50 = 70 nM T58921 COPU51 57402225 EC50 > 10000 nM T58921 CL32MT 57402244 EC50 = 310 nM T58921 C69PVW 57403073 EC50 > 5200 nM T58921 C7HKJ2 57403763 EC50 = 67 nM T58921 CXA36C 57404419 EC50 = 22600 nM T58921 CS4J1B 57404439 EC50 = 21700 nM T58921 C54ADC 57409555 EC50 = 1150 nM T58921 C4TH7G 57409556 EC50 = 11050 nM T58921 CY9CA0 58031728 IC50 = 20 nM T58921 CS6W8J 58218630 EC50 = 17000 nM T58921 CP60JL 58218638 EC50 = 32000 nM T58921 C1Y7WA 58754075 IC50 = 17.99 nM T58921 CLOJ94 58977440 EC50 = 2850 nM T58921 CT39UP 58977442 IC50 = 4280 nM T58921 CE0Y7W 58977463 IC50 = 50 nM T58921 CN6G8S 58977476 EC50 = 5650 nM T58921 CDX3L4 58977524 IC50 = 210 nM T58921 C3L2SG 58977541 EC50 = 2500 nM T58921 CW79RE 58977572 IC50 = 8110 nM T58921 CWL7J2 58977618 EC50 = 24000 nM T58921 C0A6OI 58977630 EC50 = 1060 nM T58921 C1MDW5 58977670 IC50 > 10000 nM T58921 CMTB34 58977737 IC50 = 1160 nM T58921 CIAZ23 58977763 EC50 = 10 nM T58921 CFUB93 58977773 IC50 = 590 nM T58921 CSO5C6 58977817 EC50 = 13300 nM T58921 CCS43U 58977846 IC50 = 80 nM T58921 CK6Y1Q 58977874 IC50 = 140 nM T58921 CI86BL 58977881 EC50 = 6170 nM T58921 C85QWJ 58977899 IC50 = 2830 nM T58921 C0X2IS 58977913 IC50 = 3570 nM T58921 CG1YR0 58977919 IC50 = 1530 nM T58921 CJQ4R7 59026512 EC50 = 4180 nM T58921 C4Y8DZ 59066713 IC50 > 10000 nM T58921 CP9E4V 59096898 EC50 = 19.95 nM T58921 CBQE87 59411499 EC50 = 530 nM T58921 CN9CX2 59411513 EC50 = 540 nM T58921 CE3Q2I 59411578 EC50 = 52 nM T58921 C94GHB 59835721 EC50 = 50 nM T58921 C5RH7K 60165459 EC50 = 250 nM T58921 C79PXW 60166133 EC50 > 10000 nM T58921 COCI72 60166134 EC50 > 10000 nM T58921 CO2X7F 60166264 EC50 > 10000 nM T58921 CY31AP 60166265 EC50 > 10000 nM T58921 C38XJT 60166266 EC50 > 10000 nM T58921 CFA9N8 60166267 EC50 > 10000 nM T58921 CES4D2 60166268 EC50 > 10000 nM T58921 C3P5MV 60166383 EC50 > 10000 nM T58921 CR01ID 60166384 EC50 > 10000 nM T58921 C6U3KL 60166385 EC50 > 10000 nM T58921 CN78JU 60166386 EC50 > 10000 nM T58921 C7IW2B 60166387 EC50 > 10000 nM T58921 CC3HM4 60166513 EC50 > 10000 nM T58921 CL0V6S 60166514 EC50 > 10000 nM T58921 CON53Z 60166515 EC50 > 10000 nM T58921 CU2O0N 60166516 EC50 > 10000 nM T58921 CZ8VU0 60166647 EC50 > 10000 nM T58921 CYT71B 60166648 EC50 > 10000 nM T58921 CG71ZE 60166649 EC50 > 10000 nM T58921 CC4YD6 60166650 EC50 > 10000 nM T58921 C3LGI6 60166651 EC50 > 10000 nM T58921 CALX08 60166891 EC50 > 10000 nM T58921 CD6RH2 66560742 IC50 = 650 nM T58921 C5FAY1 66561969 EC50 = 5000 nM T58921 CT3KH4 66575622 EC50 = 10000 nM T58921 C6NIF3 67072752 EC50 > 10000 nM T58921 C2RDZ8 68002585 EC50 = 30000 nM T58921 CONJ97 68159303 IC50 = 7200 nM T58921 C7T8RU 68279071 IC50 = 2000 nM T58921 C16CBO 68545524 EC50 = 6.7 nM T58921 CI5NR2 68548126 EC50 = 5.2 nM T58921 C5UV1A 68549194 EC50 = 94 nM T58921 C0CL4W 68549563 EC50 = 3.4 nM T58921 C2NDL6 68549573 EC50 = 6.2 nM T58921 CA5X0M 68549581 EC50 = 32 nM T58921 C5HR6P 68549591 EC50 > 10000 nM T58921 CVZK04 68549596 EC50 = 15 nM T58921 C9CZ6M 68549760 EC50 = 32 nM T58921 C8X9VG 68551173 EC50 = 48 nM T58921 C4LFG9 68551229 EC50 = 80 nM T58921 C75LCI 68551242 EC50 = 6.9 nM T58921 CS9WE3 68551874 EC50 = 59 nM T58921 COA24N 68552841 EC50 = 2.3 nM T58921 CX19GP 68552853 EC50 = 11 nM T58921 C3XQP8 68553004 EC50 = 1.5 nM T58921 C3U6LG 68553324 EC50 = 7.4 nM T58921 C3YBW1 68553559 EC50 = 8.6 nM T58921 CB7F3G 68553911 EC50 = 190 nM T58921 C16UXJ 68554159 EC50 > 10000 nM T58921 CPQ0T2 68554991 EC50 = 26 nM T58921 C2SVJ4 68661324 EC50 = 307 nM T58921 CF71ZG 68661359 EC50 = 550 nM T58921 C0XIR1 68661491 EC50 = 235 nM T58921 CE25MB 68661514 EC50 = 45 nM T58921 CAK3E0 68661534 EC50 = 95 nM T58921 CZ64KE 68661565 EC50 = 92 nM T58921 CGN64W 68661587 EC50 = 79 nM T58921 CXT3L7 68661602 EC50 = 39 nM T58921 C1T8YF 68661621 EC50 = 21 nM T58921 CAJV64 68661690 EC50 = 797 nM T58921 CELF49 68661767 EC50 = 139 nM T58921 CYAX75 68661771 EC50 = 845 nM T58921 C5WPA0 68661793 EC50 = 113 nM T58921 C34MPJ 68661800 EC50 = 64 nM T58921 CE9T6Z 68661809 EC50 = 23 nM T58921 C4P1LJ 68661862 EC50 = 12400 nM T58921 CYD08V 68661925 EC50 = 50 nM T58921 CC1W7Z 68661980 EC50 = 90 nM T58921 CNJA68 68661986 EC50 = 41 nM T58921 C6NEB4 68662059 EC50 = 143 nM T58921 CF57AT 68662065 EC50 = 22 nM T58921 C81RYD 68662112 EC50 = 1434 nM T58921 C0MA7X 68662132 EC50 = 299 nM T58921 CS5K4W 68662136 EC50 = 4.4 nM T58921 CBA7H4 68662161 EC50 = 86 nM T58921 CV1LZ7 68662186 EC50 = 56 nM T58921 CT18SJ 68662238 EC50 = 122 nM T58921 CURO91 68662593 EC50 = 6094 nM T58921 C1WL3P 68674744 EC50 = 1558 nM T58921 CKM6E9 68675602 EC50 = 910 nM T58921 CS4V7A 68676158 EC50 = 153 nM T58921 C9PF1U 68676459 EC50 = 378 nM T58921 CH62WK 68676471 EC50 = 55 nM T58921 CM1O9L 68676633 EC50 = 72 nM T58921 CE9IP3 68676761 EC50 = 265 nM T58921 CI7DX4 68676782 EC50 = 175 nM T58921 C93PTK 68676826 EC50 = 35 nM T58921 CFN69J 68677403 EC50 = 284 nM T58921 CIYO07 68677705 EC50 > 5000 nM T58921 CIU96H 68677842 EC50 = 206 nM T58921 C8ML2B 69016303 EC50 = 251 nM T58921 CFKV51 69078165 EC50 = 320 nM T58921 CZ3WJ6 70680568 EC50 = 1000 nM T58921 CRQU32 70681335 EC50 = 290 nM T58921 C4M7WJ 70681370 EC50 = 61 nM T58921 CLC72I 70681461 EC50 = 3.1 nM T58921 CY9GZ8 70681800 IC50 = 5.998 nM T58921 C2DZ3G 70681801 IC50 = 2238.72 nM T58921 CSEF42 70681805 IC50 = 139 nM T58921 CMT6J3 70681806 IC50 = 449.78 nM T58921 C3A0DO 70682526 IC50 > 60000 nM T58921 CLJU20 70682537 IC50 > 60000 nM T58921 C2SVR8 70682538 IC50 > 60000 nM T58921 C15AQZ 70683585 EC50 = 10 nM T58921 CB4A7U 70683915 IC50 = 289.73 nM T58921 CG40IU 70684617 IC50 > 60000 nM T58921 CO1MQ8 70684618 IC50 > 60000 nM T58921 CU5VH3 70684619 IC50 = 30200 nM T58921 CDI86Q 70685690 EC50 > 10000 nM T58921 C7TJC3 70686048 IC50 = 128 nM T58921 C13CJK 70686054 IC50 = 1059.25 nM T58921 CVK46F 70686763 IC50 > 60000 nM T58921 CWJ6U3 70686764 IC50 > 60000 nM T58921 CCBM25 70688041 IC50 = 900 nM T58921 CEL43F 70688075 EC50 > 10000 nM T58921 C40KCB 70688165 IC50 = 6095.37 nM T58921 CFY6Z4 70688166 IC50 = 479.73 nM T58921 CP72KL 70688172 IC50 = 7998.34 nM T58921 C70SIB 70688836 IC50 > 60000 nM T58921 C0NG7E 70689734 EC50 = 38 nM T58921 CYJ75M 70690069 IC50 = 540 nM T58921 CIC8V5 70690196 IC50 = 59.02 nM T58921 CLF25D 70690926 IC50 > 60000 nM T58921 CB3ZC2 70690927 IC50 > 60000 nM T58921 C6FA0H 70690939 IC50 > 60000 nM T58921 C69MGD 70692364 IC50 = 1499.68 nM T58921 C34KXB 70692371 IC50 = 62.95 nM T58921 C90XVL 70693065 IC50 > 60000 nM T58921 CC2EK8 70693080 IC50 > 60000 nM T58921 CR2YQ9 70693621 EC50 = 52300 nM T58921 C90MIS 70694287 IC50 = 890 nM T58921 C5C9HR 70694419 IC50 = 30 nM T58921 C4DRC8 70694428 IC50 = 29.99 nM T58921 C29DRB 70694429 IC50 = 19.01 nM T58921 C2WC4V 70695111 IC50 > 60000 nM T58921 C92QMH 70695112 IC50 > 60000 nM T58921 CMNE57 70695113 IC50 > 60000 nM T58921 CV3T4P 70695727 EC50 = 48700 nM T58921 CR2PJ4 70695728 EC50 = 18900 nM T58921 CI20AZ 70696193 EC50 = 5.5 nM T58921 CBSY90 70696194 EC50 > 10000 nM T58921 CIZ7O3 70696377 EC50 = 6000 nM T58921 CL0JN8 70696489 IC50 = 4102.04 nM T58921 C90GXS 70696490 IC50 = 399.02 nM T58921 CTQ37A 70697163 IC50 > 60000 nM T58921 CG60YB 71074285 EC50 = 129 nM T58921 C0GHQ3 71074396 EC50 = 3 nM T58921 CDO46S 71074518 IC50 = 0.54 nM T58921 C6BR8G 71074647 IC50 = 14 nM T58921 CMY0L9 71074661 EC50 = 124 nM T58921 CY2VU8 71074698 IC50 = 3 nM T58921 C7XS9K 71074707 IC50 = 21 nM T58921 C3YR5S 71074714 IC50 = 20 nM T58921 CD0P3A 71074731 Ki = 12 nM T58921 C6ZW1C 71074744 IC50 = 1 nM T58921 CB17LH 71074807 IC50 = 5 nM T58921 CSPJ87 71074820 EC50 = 179 nM T58921 CVC9X6 71074842 IC50 = 6 nM T58921 CQ26DN 71074844 IC50 = 6 nM T58921 C4TNR2 71074846 EC50 = 5665 nM T58921 C6AP1O 71074861 IC50 = 38 nM T58921 C06VNX 71074894 IC50 = 1 nM T58921 C2SD9N 71074907 Ki = 244 nM T58921 C2S0EB 71074929 EC50 = 47 nM T58921 CLSX16 71074982 EC50 = 14 nM T58921 CK36UL 71075168 EC50 = 1 nM T58921 C1R2MS 71075179 IC50 = 0.9 nM T58921 C1ZP9L 71075304 EC50 = 363 nM T58921 CT29FZ 71075689 EC50 = 4907 nM T58921 C9PA6Y 71449654 EC50 = 33100 nM T58921 CL8W1E 71450437 EC50 = 890 nM T58921 CDVK19 71450438 EC50 = 670 nM T58921 CZO16C 71450439 EC50 > 25000 nM T58921 CK5WV7 71450440 EC50 = 1300 nM T58921 C2EUK6 71450447 EC50 = 5800 nM T58921 CC5T1Z 71450448 EC50 = 1400 nM T58921 CPS54B 71450449 EC50 = 800 nM T58921 CGN2A9 71452269 EC50 = 330 nM T58921 CQY90O 71452270 EC50 > 25000 nM T58921 CAR5V4 71452275 EC50 = 7900 nM T58921 C9DX5U 71452276 EC50 = 800 nM T58921 CSN6G2 71452725 EC50 = 1566 nM T58921 C9ERN1 71453290 EC50 > 50000 nM T58921 CP27KN 71454069 EC50 = 700 nM T58921 CT27RV 71454077 EC50 = 6000 nM T58921 C5US2A 71455005 EC50 > 50000 nM T58921 CU34JE 71455800 EC50 = 310 nM T58921 CRQA20 71455801 EC50 = 2200 nM T58921 CA2L9V 71455810 EC50 = 6900 nM T58921 CIZA80 71455811 EC50 = 5900 nM T58921 C98QRS 71457369 EC50 = 6000 nM T58921 CJ5WR8 71457584 EC50 = 180 nM T58921 C4O7MV 71457585 EC50 = 71 nM T58921 CU49YK 71457599 EC50 = 21000 nM T58921 CM4F2S 71457600 EC50 = 39300 nM T58921 C9GET3 71458051 Ki = 1330 nM T58921 CRF20V 71458052 EC50 = 1195 nM T58921 C16BJE 71459228 EC50 = 2000 nM T58921 CC17GK 71459487 EC50 = 42 nM T58921 CP64MJ 71459495 EC50 = 54600 nM T58921 CWO9U1 71459496 EC50 = 800 nM T58921 C4EB3N 71459497 EC50 = 10000 nM T58921 C1FP8C 71461220 EC50 = 4.7 nM T58921 CQW65K 71461221 EC50 = 16000 nM T58921 CDLM36 71461229 EC50 = 5400 nM T58921 CL2EG1 71461230 EC50 = 75200 nM T58921 C0ZM1O 71461231 EC50 = 12600 nM T58921 C6O0TB 71462957 EC50 = 7700 nM T58921 CAH63D 71462958 EC50 > 25000 nM T58921 CY6A5T 71462959 EC50 = 8800 nM T58921 CTCS46 71462964 EC50 = 32000 nM T58921 CS65PB 71478598 EC50 = 2532 nM T58921 CA95RY 71520500 EC50 = 42 nM T58921 CGTO05 71520501 EC50 = 295 nM T58921 CQ80JF 71521194 EC50 > 100000 nM T58921 CC3F8V 71521195 EC50 > 100000 nM T58921 CP4W1D 71521196 EC50 = 1250 nM T58921 CHN49X 71521298 EC50 > 100000 nM T58921 C94MCT 71521299 EC50 = 1710 nM T58921 C9C2NZ 71521300 EC50 = 942 nM T58921 CM79CL 71521301 EC50 = 103 nM T58921 CO01SV 71521302 EC50 = 97 nM T58921 C5V9UO 71521416 EC50 = 685 nM T58921 C89DQL 71521417 EC50 = 187 nM T58921 CAT53R 71521418 EC50 = 20 nM T58921 CJU56D 71521419 EC50 = 159 nM T58921 CM96IV 71521503 EC50 = 108 nM T58921 CFA2P7 71521504 EC50 = 449 nM T58921 CGN94D 71521505 EC50 = 3580 nM T58921 CA0K3Z 71521506 EC50 = 3640 nM T58921 CW1G9U 71521507 EC50 > 25000 nM T58921 CPC40O 71521585 EC50 = 4470 nM T58921 C9JQ3C 71525043 EC50 = 30 nM T58921 CLX4U0 71525044 EC50 = 15 nM T58921 CHX52K 71525045 EC50 = 30 nM T58921 CLC2I8 71525046 EC50 = 15 nM T58921 C9R8KL 71525047 EC50 = 20 nM T58921 CG3NY8 71525048 IC50 = 160 nM T58921 COR5V4 71525086 IC50 = 49 nM T58921 C9WL8K 71525087 IC50 > 10000 nM T58921 C4Y1UF 71525166 IC50 > 10000 nM T58921 C4Z0YK 71525167 EC50 = 30 nM T58921 C3QKM9 71525168 EC50 = 100 nM T58921 CNFJ29 71525169 IC50 = 27 nM T58921 CD26MN 71525170 EC50 = 90 nM T58921 C06DJE 71525218 IC50 = 32 nM T58921 C1OF9Y 71525219 EC50 = 300 nM T58921 C83BHF 71525220 EC50 = 100 nM T58921 C9KRS5 71525221 IC50 = 40 nM T58921 C5VG9H 71525222 EC50 = 250 nM T58921 CJE5P1 71525223 IC50 = 30 nM T58921 COC18S 71525259 EC50 = 2000 nM T58921 CO64EH 71544680 EC50 = 590 nM T58921 C0AV4J 71544681 EC50 = 460 nM T58921 C72FAV 71544682 EC50 = 1360 nM T58921 CS56TM 71544683 EC50 = 640 nM T58921 CJ93XY 71544684 EC50 = 690 nM T58921 CKTE38 71544685 EC50 = 1000 nM T58921 C9BXE3 71544686 EC50 = 1400 nM T58921 CLS10T 71544851 EC50 = 2300 nM T58921 C3GWQ1 71544852 EC50 = 1200 nM T58921 CFZ3A6 71547107 EC50 = 700 nM T58921 CT0ZA3 71547108 EC50 = 700 nM T58921 COVC32 71547109 EC50 = 3100 nM T58921 C4W5PD 71547110 EC50 = 2040 nM T58921 C6FZ7C 71547111 EC50 = 2540 nM T58921 CLE7O6 71582884 EC50 = 713.9 nM T58921 C8JC1N 71582885 EC50 = 3095 nM T58921 CAK2X1 71584600 EC50 = 102.6 nM T58921 CI5UP1 71584601 EC50 = 186.1 nM T58921 C19HFD 71584602 EC50 = 844 nM T58921 CQ35BM 71584603 EC50 = 1688 nM T58921 CL4A2V 71604423 EC50 = 16 nM T58921 C10SPC 71616170 EC50 = 19 nM T58921 CNPK13 71616171 EC50 = 110 nM T58921 CI1LF2 71616173 EC50 = 20 nM T58921 C9U6VX 71616290 EC50 = 34 nM T58921 CK58CF 71616294 EC50 = 39 nM T58921 C6LT3W 71616409 EC50 = 72 nM T58921 C2EK8O 71712902 IC50 = 62700 nM T58921 CRS79L 71712906 IC50 = 38700 nM T58921 CSHD03 71713038 IC50 = 56200 nM T58921 C7EX4R 71718932 EC50 = 600 nM T58921 C5NU0T 71721539 IC50 = 15000 nM T58921 CMFD46 72734874 EC50 = 6400 nM T58921 C2K0GM 72734875 EC50 = 7600 nM T58921 CBO3D4 72734876 EC50 = 3900 nM T58921 C6WKI3 72735052 EC50 = 5700 nM T58921 C3QIV9 72735053 EC50 = 7200 nM T58921 C4TLU8 72735056 EC50 = 1300 nM T58921 CWHB65 72735057 EC50 = 2900 nM T58921 CZB62X 72735237 EC50 = 3600 nM T58921 CU07KO 72735238 EC50 = 3400 nM T58921 CKH6N5 72735239 EC50 = 4100 nM T58921 CF8N6W 72735417 EC50 = 2300 nM T58921 CX2ND4 72735418 EC50 = 3800 nM T58921 C4JSP6 72735591 EC50 = 3700 nM T58921 CFW41I 73167563 EC50 = 120 nM T58921 CX20AE 73347299 EC50 = 912.01 nM T58921 CBSQ86 73347300 EC50 = 1659.59 nM T58921 C1GIP0 73347301 EC50 = 1258.93 nM T58921 CUZC61 73347302 EC50 = 8912.51 nM T58921 C0VHS6 73351898 EC50 = 7079.46 nM T58921 C93SWK 73351899 EC50 = 1584.89 nM T58921 CUEA53 73356438 EC50 = 316.23 nM T58921 C57URV 76309038 EC50 = 0.1 nM T58921 C8X4IT 76309039 EC50 = 23.99 nM T58921 C35STH 76310606 EC50 = 2650 nM T58921 C18EZQ 76310607 EC50 = 2 nM T58921 C7DE3L 76310608 EC50 = 90 nM T58921 CIR72S 76310609 EC50 = 130 nM T58921 C7IOX1 76310610 EC50 = 640 nM T58921 C49IUW 76311770 EC50 = 31.62 nM T58921 C82WBS 76311981 EC50 = 12000 nM T58921 CAV64K 76312305 EC50 = 8000 nM T58921 CJ4P7G 76312720 EC50 = 1.288 nM T58921 C5X3HV 76312721 EC50 = 0.3388 nM T58921 C41CED 76315850 EC50 = 11000 nM T58921 C9QN4E 76317814 EC50 = 350 nM T58921 CP7E1N 76317815 EC50 = 180 nM T58921 CGT93D 76319009 EC50 = 1 nM T58921 C75YZJ 76319010 EC50 = 630.96 nM T58921 C4SW3D 76319206 EC50 = 167 nM T58921 CB19YJ 76319208 EC50 = 106 nM T58921 CF9C8Z 76319552 EC50 = 9000 nM T58921 C32YPJ 76321033 EC50 = 23 nM T58921 CD36HB 76321525 EC50 = 80 nM T58921 C7UCQ8 76322858 EC50 = 47 nM T58921 CR12QV 76325125 EC50 = 6 nM T58921 CH1W8N 76325126 EC50 = 390 nM T58921 C9G1TZ 76326728 EC50 = 10000 nM T58921 C2GY6R 76328690 EC50 = 280 nM T58921 C5F4EM 76330047 EC50 = 27 nM T58921 CQ3SY4 76330398 EC50 = 9000 nM T58921 C78XLM 76330830 EC50 = 0.7079 nM T58921 CT65IA 76333688 EC50 = 23 nM T58921 CR6AG1 76334423 EC50 = 19.95 nM T58921 CIW0C8 76334424 EC50 = 4.677 nM T58921 CFY25B 76335715 IC50 > 25000 nM T58921 CPT9V0 77845055 EC50 > 50000 nM T58921 CH0A1L 78319338 EC50 = 0.38 nM T58921 CBA6J1 78319339 EC50 = 183 nM T58921 C6X5MD 86279340 EC50 = 5500 nM T58921 C5WG3I 86582930 EC50 = 1622 nM T58921 C63WUO 87537807 EC50 = 41 nM T58921 CH4A7L 88928909 IC50 = 8460 nM T58921 CU29QZ 90159227 EC50 = 2600 nM T58921 CL2R0D 90466288 IC50 = 14700 nM T58921 CTBQ27 90469357 EC50 = 1298 nM T58921 CR3I0E 90469358 EC50 > 100000 nM T58921 CY09NA 90469423 EC50 > 100000 nM T58921 C0GQ9R 90469424 EC50 > 100000 nM T58921 CSRZ25 90469425 EC50 > 100000 nM T58921 CN17FZ 90644288 EC50 > 10000 nM T58921 CI2Q9P 90656006 EC50 = 21000 nM T58921 CD79FV 90656011 EC50 = 18100 nM T58921 CY59UG 90656014 EC50 = 26000 nM T58921 C4BA8W 90656430 IC50 > 100000 nM T58921 CR21SD 90676722 EC50 = 13000 nM T58921 CXMC90 90676723 EC50 = 37000 nM T58921 CKJ89N 90676724 EC50 = 23000 nM T58921 CYJR07 90676727 EC50 = 41000 nM T58921 CA9PL8 91663316 IC50 = 21300 nM T58921 CI92WR 91664317 IC50 = 650 nM T58921 C7R6IK 101882290 EC50 = 2990 nM T58921 C73YEJ 101889825 EC50 = 1700 nM T58921 C7X5DQ 101889826 EC50 = 1900 nM T58921 C4C3MB 101889827 EC50 = 2000 nM T58921 C9JT3G 101889828 EC50 = 1700 nM T58921 CM1U8G 101889829 EC50 = 1200 nM T58921 CE74QT 101896434 EC50 = 6300 nM T58921 CCW4S0 101896435 EC50 = 5000 nM T58921 CA6I4Y 101896436 EC50 = 2600 nM T58921 CFCE51 101896437 EC50 = 18000 nM T58921 C8CJR5 102004339 EC50 > 100000 nM T58921 CQLI09 102313441 EC50 = 6.7 nM T58921 CKQ89B 102313442 EC50 = 6.7 nM T58921 C18LMP 102313443 EC50 = 1.9 nM T58921 C1CN0A 117629817 EC50 > 10000 nM T58921 CYQ36G 117953851 IC50 > 10000 nM T58921 CS0G6T 117964950 IC50 = 1100 nM T58921 C1WM4V 117964951 IC50 > 10000 nM T58921 C2KJH5 117964960 IC50 = 1800 nM T58921 C4S9EM 117964962 IC50 = 320 nM T58921 C9AW4X 117964963 IC50 = 9100 nM T58921 CS4GJ9 117964973 IC50 = 1300 nM T58921 CDXK37 117964975 IC50 = 3400 nM T58921 CN6RT8 117964978 IC50 = 1500 nM T58921 C0KL3C 117964989 IC50 = 2100 nM T58921 C96BSK 117964998 IC50 = 760 nM T58921 CW27MY 118063735 EC50 > 10000 nM T58921 C0O8HY 118708437 EC50 = 38.9 nM T58921 C25FLM 118708438 EC50 = 7 nM T58921 C95BSE 118708439 EC50 = 10.4 nM T58921 C1CWS6 118708440 EC50 = 2.2 nM T58921 CCLN05 118708441 EC50 = 5.3 nM T58921 CTWH29 118708442 EC50 = 11.7 nM T58921 CT7ZN0 118708443 EC50 = 2.2 nM T58921 C2B0NR 118708577 EC50 = 12400 nM T58921 CS9L7H 118708578 EC50 = 1060 nM T58921 CVHW16 118708579 EC50 = 690 nM T58921 C1K9RV 118708580 EC50 = 1200 nM T58921 CIU9H3 118708581 EC50 = 2360 nM T58921 C1C6RK 118708582 EC50 = 490 nM T58921 CT4RD5 118714597 EC50 = 3900 nM T58921 C9M7RL 118714598 EC50 = 8500 nM T58921 C49HBU 118714599 EC50 = 4500 nM T58921 C5U4QT 118714600 EC50 = 25000 nM T58921 CN4PU6 118714603 EC50 = 6900 nM T58921 CFVY93 118714604 EC50 = 11000 nM T58921 CA1RT3 118714624 EC50 = 6200 nM T58921 C8AS1X 118714625 EC50 = 5000 nM T58921 CGI3J6 118714626 EC50 = 13500 nM T58921 CB27OT 118714627 EC50 = 4500 nM T58921 CP10TG 118714628 EC50 = 5800 nM T58921 C98ILP 118714629 EC50 = 1900 nM T58921 C0X3NL 118714630 EC50 = 4400 nM T58921 C7KS6D 118714631 EC50 = 5400 nM T58921 CR7I1H 118714632 EC50 = 6300 nM T58921 CL1VI2 118714636 EC50 = 5400 nM T58921 CNA46V 118714637 EC50 = 9000 nM T58921 C0PTU8 118720593 EC50 = 25000 nM T58921 CY0L3P 118721127 EC50 = 12 nM T58921 CUY8C6 118721128 EC50 = 47 nM T58921 CF6K3L 118721129 EC50 = 26 nM T58921 C09GZO 118721130 EC50 = 12 nM T58921 C04OPW 118721131 EC50 = 21 nM T58921 CFCN47 118721132 EC50 = 84 nM T58921 CR41YO 118721133 EC50 = 32 nM T58921 C0XS6T 118721134 EC50 = 183 nM T58921 C8EZX7 118721135 EC50 = 1370 nM T58921 CVC60I 118721136 EC50 = 39 nM T58921 CIWK60 118721137 EC50 = 47 nM T58921 CIAE91 118721138 EC50 = 29 nM T58921 CZT5N2 118721140 EC50 = 250 nM T58921 CNL01R 118721141 EC50 = 640 nM T58921 C5Y9BH 118722565 IC50 = 5000 nM T58921 CZP8E7 118725344 EC50 = 4700 nM T58921 CKC50A 118725345 EC50 = 8700 nM T58921 C5ENC7 118725346 EC50 = 9400 nM T58921 CTH73Y 118725347 EC50 = 6900 nM T58921 CQ4OY5 118725348 EC50 = 17400 nM T58921 C9M1BC 118725349 EC50 = 4400 nM T58921 CF3LH1 118726796 EC50 = 43000 nM T58921 C4URP2 118726797 EC50 = 28000 nM T58921 CNRJ62 118726798 EC50 = 12800 nM T58921 CSM7R4 118726800 EC50 = 7900 nM T58921 CG6Y7T 118726801 EC50 = 3800 nM T58921 C46WTE 118726802 EC50 = 3650 nM T58921 CSV2H4 118726804 EC50 = 5600 nM T58921 CJ2BR5 118726806 EC50 = 4500 nM T58921 C6YJQ9 118726808 EC50 = 2100 nM T58921 C2G5WT 118726809 EC50 = 1800 nM T58921 C92FYQ 118726811 EC50 = 1250 nM T58921 CC7A0V 118726812 EC50 = 9400 nM T58921 C4T1FZ 118726813 EC50 = 12400 nM T58921 C7UKX3 118726814 EC50 = 1000 nM T58921 C92IJW 118726815 EC50 = 680 nM T58921 C2FWY0 118726937 EC50 = 720 nM T58921 C6XH0K 118726938 EC50 = 11700 nM T58921 CE7L6H 118726939 EC50 = 12900 nM T58921 CB23OM 118726943 EC50 = 5170 nM T58921 CVU2B8 118726944 EC50 = 2110 nM T58921 C7EU9N 118726945 EC50 = 4640 nM T58921 CXEG20 118726946 EC50 = 2560 nM T58921 CY3J0G 118726949 IC50 = 4300 nM T58921 C4J5EW 118726952 EC50 = 3770 nM T58921 CVO6Y5 118726954 EC50 = 1260 nM T58921 CA8TS2 118726955 EC50 = 2160 nM T58921 COS6Z5 118727475 EC50 > 32000 nM T58921 C9OTJ4 118727476 EC50 = 4180 nM T58921 CC2JU8 118727477 IC50 = 240 nM T58921 CUW31A 118727478 EC50 = 9680 nM T58921 CML56Z 118727479 IC50 = 1820 nM T58921 CF0YU2 118727480 IC50 > 10000 nM T58921 CI1H5O 118727481 IC50 = 110 nM T58921 C5AO7P 118727482 IC50 = 520 nM T58921 C8EC2D 118727483 IC50 = 1590 nM T58921 C2F1AI 118727484 IC50 = 340 nM T58921 C4E3AX 121269371 EC50 > 10000 nM T58921 CW23RD 121269378 EC50 > 10000 nM T58921 C3AP2B 121269382 EC50 > 10000 nM T58921 CX4AN2 121269406 EC50 > 10000 nM T58921 CLRU83 121269424 EC50 > 10000 nM T58921 CC32JH 121277016 EC50 > 10000 nM T58921 C0BKL7 121277018 EC50 > 10000 nM T58921 CE3YL2 121277093 EC50 > 10000 nM T58921 CPA8J7 121277097 EC50 > 10000 nM T58921 C6TBD2 121345502 EC50 > 20000 nM T58921 CB0P3T 122179683 EC50 = 155 nM T58921 C8B1KR 122179686 Ki = 440 nM T58921 CPT38B 122179687 IC50 = 190 nM T58921 CLR57W 122182699 IC50 > 10000 nM T58921 CPJ3M7 122182700 IC50 = 5600 nM T58921 CK5WJ9 122182701 IC50 = 2900 nM T58921 CY0M6P 122182702 IC50 = 7700 nM T58921 CLV91R 122182703 IC50 = 5500 nM T58921 C0BI8N 122183534 EC50 = 1900 nM T58921 CHYL24 122183546 EC50 = 1300 nM T58921 CHUW19 122184171 IC50 = 4200 nM T58921 CFMX82 122184177 IC50 > 10000 nM T58921 CNV03S 122189255 IC50 = 4000 nM T58921 C40QCP 125623112 EC50 > 100000 nM T58921 CH0UW8 126970815 EC50 = 131 nM T58921 C6R8QV 127035275 IC50 = 17 nM T58921 CI8RG4 127035427 EC50 = 100 nM T58921 CKV27T 127035467 IC50 = 10100 nM T58921 C9Y6NA 127036555 IC50 > 200000 nM T58921 CJ7AQ1 127037232 IC50 = 6500 nM T58921 C2R3LT 127037251 IC50 = 84000 nM T58921 CN3SG4 127037377 IC50 = 78400 nM T58921 CW1JT2 127037542 IC50 = 59100 nM T58921 C8RMJ9 127037543 IC50 = 191000 nM T58921 C1P5EV 127037556 IC50 = 22200 nM T58921 C4RP2D 127038538 EC50 = 11000 nM T58921 C4GZ1S 127039678 EC50 = 4000 nM T58921 CG1S6F 127039682 EC50 = 3500 nM T58921 C9OVT1 127039683 EC50 = 8000 nM T58921 C8VXT4 127040583 EC50 = 1800 nM T58921 C7XV1H 127040584 EC50 = 4800 nM T58921 CVQT15 127040585 EC50 = 2200 nM T58921 CN45YE 127041516 EC50 = 4200 nM T58921 C39LHD 127041523 EC50 = 6400 nM T58921 C8ZQT1 127041821 EC50 = 8000 nM T58921 C3B6SN 127041822 EC50 = 3000 nM T58921 C82RIP 127042123 EC50 = 6300 nM T58921 C9H3DO 127042124 EC50 = 3000 nM T58921 C7J8AO 127042143 EC50 = 1400 nM T58921 C54WUI 127042144 EC50 = 300 nM T58921 C3I1BC 127042145 EC50 = 2800 nM T58921 COUD73 127042146 EC50 = 600 nM T58921 CRN48C 127042147 EC50 = 2000 nM T58921 C74HEQ 127042148 EC50 = 300 nM T58921 C10ZDF 127042456 EC50 = 2000 nM T58921 C91VBI 127042458 EC50 = 7000 nM T58921 C3SFH0 127042459 EC50 = 4000 nM T58921 C40UWZ 127042480 EC50 = 900 nM T58921 C3X0VB 127042481 EC50 = 1500 nM T58921 C1RZE5 127042482 EC50 = 2000 nM T58921 C9I0GA 127042483 EC50 = 3000 nM T58921 CAC1X8 127042485 EC50 = 16000 nM T58921 C45JCU 127042486 EC50 = 13500 nM T58921 C3PYC8 127043494 EC50 = 4383 nM T58921 C19YRU 127043495 EC50 = 1235 nM T58921 CP2GI3 127043496 EC50 = 1504 nM T58921 C4EZC8 127043497 EC50 = 1255 nM T58921 C1BI8N 127043498 EC50 = 1087 nM T58921 C5WP3T 127043675 EC50 = 2062 nM T58921 CQ72PD 127043676 EC50 = 2384 nM T58921 CD0Q6O 127043844 EC50 = 414 nM T58921 CQ1O2V 127043845 EC50 > 25000 nM T58921 CIB59P 127043846 EC50 = 4273 nM T58921 C5D7PK 127043847 EC50 = 2013 nM T58921 CP83SU 127044158 EC50 = 9168 nM T58921 C5YL1I 127044159 EC50 = 2857 nM T58921 C3Z2WU 127044160 EC50 = 10010 nM T58921 CZ2GY0 127044161 EC50 = 8607 nM T58921 CLYV46 127044284 EC50 = 2182 nM T58921 CG1RN9 127051847 EC50 = 6000 nM T58921 CL56FH 129147662 IC50 = 4480 nM T58921 CNB6Y7 130417522 EC50 = 11100 nM T58921 CDV84X 131747741 EC50 > 20000 nM T58921 CBXG19 132606863 EC50 = 4400 nM T58921 CTC10K 132609296 IC50 = 371 nM T58921 CLQG26 132609297 IC50 = 350 nM T58921 C2MY7T 132609298 IC50 = 369 nM T58921 C52SHY 132609299 IC50 = 402 nM T58921 C2SJR7 132609300 IC50 = 464 nM T58921 C51EAL 132609301 IC50 = 353 nM T58921 C21RJM 132609302 IC50 = 980 nM T58921 C4HYA2 132609303 IC50 = 590 nM T58921 C5WF9I 132961628 IC50 = 4000 nM T58921 CMO0Y4 132961629 IC50 = 482 nM T58921 CV1HP6 132961630 IC50 = 4000 nM T58921 C5M4KG 132961631 IC50 = 350 nM T58921 C6SUZ1 134132400 EC50 = 8030 nM T58921 CJ4W1X 134136024 EC50 = 840 nM T58921 CA0KZ8 134138434 EC50 = 3150 nM T58921 CG9IH6 134142790 EC50 = 1860 nM T58921 C0QX9P 134146293 IC50 = 1320 nM T58921 C9BXT3 134146519 IC50 = 369 nM T58921 CC7SD3 134146881 EC50 = 6240 nM T58921 C53NKB 134146909 IC50 = 1150 nM T58921 COU0X5 134151475 EC50 = 170 nM T58921 CA90GO 134151878 IC50 = 1141 nM T58921 CRT73V 134152006 IC50 = 4000 nM T58921 C76LYZ 134152589 EC50 = 1880 nM T58921 CX47MQ 134152810 EC50 = 3060 nM T58921 CB5CD6 134156037 EC50 = 210 nM T58921 CV8IF2 134156437 IC50 = 1293 nM T58921 C98MDE 134156986 EC50 = 1050 nM T58921 CY5WF7 134157295 EC50 = 3900 nM T58921 CH0D8R 134216618 EC50 = 3.3 nM T58921 CGX6K0 135444763 EC50 = 9800 nM T58921 CV6OP5 135513372 EC50 > 10000 nM T58921 CK04WX 135567387 EC50 = 2.4 nM T58921 CL6Q7I 136000613 EC50 = 14600 nM T58921 CYXD83 136036579 IC50 = 2050 nM T58921 C9IU2J 136088972 IC50 = 48 nM T58921 CBJ89X 136264026 EC50 = 2.5 nM T58921 CN7RH8 136264517 EC50 = 3.981 nM T58921 C5HWO9 136265679 EC50 = 17 nM T58921 CV1X2M 136265684 EC50 = 2.7 nM T58921 C4MZP2 136364662 EC50 = 84 nM T58921 C98FSH 136364739 EC50 = 177 nM T58921 CFQ4S1 136376542 EC50 = 166 nM T58921 CT0CR4 136376560 EC50 = 151 nM T58921 C2YDH9 136376567 EC50 = 57 nM T58921 CP47IH 136376580 EC50 = 593 nM T58921 CKW6J9 136397795 EC50 = 7 nM T58921 C2O6DI 136491120 EC50 = 5.3 nM T58921 C2MV9Q 136491135 EC50 = 1.7 nM T58921 CN0O5B 136491139 EC50 = 3 nM T58921 C9AD0I 136591472 EC50 = 2 nM T58921 CGC84N 136591486 EC50 = 1 nM T58921 C5GI3J 136591510 EC50 = 32 nM T58921 C57XVB 136591522 EC50 = 1 nM T58921 CU39XG 136591535 EC50 = 4.5 nM T58921 C6FN2L 136591583 EC50 = 1.4 nM T58921 CW8QT1 137527725 EC50 = 1730 nM T58921 CG45OX 137532803 EC50 = 7360 nM T58921 C67URH 137532805 EC50 = 1660 nM T58921 CAD2P3 137631891 EC50 = 14700 nM T58921 COTP43 137632174 EC50 = 1390 nM T58921 C7DS5O 137633219 EC50 = 147 nM T58921 CYG4I2 137633420 EC50 = 256 nM T58921 C8LBM9 137633766 EC50 = 1250 nM T58921 C68SZA 137634330 EC50 > 10000 nM T58921 C3EN2L 137634371 EC50 = 151 nM T58921 C4WR2S 137635023 EC50 = 957 nM T58921 CGUF20 137635167 EC50 = 1600 nM T58921 CU7C0K 137637447 EC50 = 3314 nM T58921 C15XNC 137637824 EC50 = 629 nM T58921 CZT6M4 137637905 EC50 = 290 nM T58921 C6LI3N 137637955 EC50 = 82 nM T58921 C69SXT 137638058 EC50 = 5810 nM T58921 C01SRK 137638871 EC50 = 169 nM T58921 C8FZ6W 137639177 EC50 = 18000 nM T58921 CI5ER2 137639724 EC50 = 201 nM T58921 CKXQ78 137640612 EC50 = 280 nM T58921 C9J0IE 137640656 EC50 = 600 nM T58921 CSP9K7 137641115 EC50 = 75 nM T58921 C75CGO 137642891 EC50 = 1350 nM T58921 CS82BE 137643489 EC50 = 1248 nM T58921 CGS98B 137643812 EC50 = 770 nM T58921 CQN59G 137643813 EC50 = 820 nM T58921 C0Z9NE 137644153 EC50 = 3400 nM T58921 CCW0B2 137644269 EC50 > 5000 nM T58921 C9N0JP 137645369 EC50 = 134 nM T58921 CZ9U8P 137646175 IC50 = 408 nM T58921 C29IKU 137646877 EC50 = 1150 nM T58921 CBC61V 137647253 EC50 = 16 nM T58921 C93IRA 137648584 EC50 = 65 nM T58921 CM76LD 137649352 EC50 = 290 nM T58921 CW7YR0 137649652 EC50 = 94 nM T58921 CVB69P 137649932 EC50 = 360 nM T58921 C0LWS1 137650297 EC50 = 930 nM T58921 CRB9Z7 137651528 EC50 = 417 nM T58921 CHQ08L 137653711 EC50 = 300 nM T58921 CFI68P 137653903 EC50 > 10000 nM T58921 CLQ48M 137654269 EC50 = 1010 nM T58921 CP3K6L 137654393 EC50 = 53 nM T58921 CS43WD 137654739 EC50 = 277 nM T58921 C7KP3N 137654758 EC50 = 2 nM T58921 CDW90U 137655271 EC50 = 410 nM T58921 CZ84GI 137655707 EC50 = 284 nM T58921 C73KNP 137656170 EC50 = 1010 nM T58921 CWVL96 137657634 EC50 = 2980 nM T58921 CBM79V 137658450 EC50 = 4090 nM T58921 C46QHL 137659090 EC50 = 4 nM T58921 CGP3J1 137659100 EC50 = 290 nM T58921 CL1RG9 137659246 EC50 = 573 nM T58921 CUOL07 137659478 EC50 = 4289 nM T58921 CU1NM2 137661255 EC50 = 190 nM T58921 C9PA8G 138911343 EC50 = 280 nM T58921 CC5X3V 139501076 EC50 = 18300 nM T58921 CFM9U6 139501078 EC50 > 100000 nM T58921 C5WRM9 139501186 EC50 > 100000 nM T58921 C9KYQ5 139501208 EC50 = 5600 nM T58921 C35EGB 141511142 EC50 = 5190 nM T58921 C95BLC 141511161 EC50 = 3670 nM T58921 CZI51H 141511162 EC50 = 910 nM T58921 CTH4W2 141511167 EC50 = 56710 nM T58921 C7KD9N 142533975 EC50 = 3100 nM T58921 CH0SV7 142534021 EC50 = 1000 nM T58921 C78UCE 142534055 EC50 = 2250 nM T58921 CEM37U 142534134 EC50 = 10300 nM T58921 CJE36P 142534202 EC50 = 1530 nM T58921 C60TYD 142738546 EC50 = 56900 nM T58921 CI0E6S 142738567 EC50 = 2400 nM T58921 C6I2JS 142738569 EC50 = 236400 nM T58921 CKS10N 145704693 EC50 = 1.6 nM T58921 CF96VY 145714275 IC50 = 99300 nM T58921 CT73UW 145949449 EC50 = 808 nM T58921 CL65HC 145949618 EC50 = 340 nM T58921 COKZ54 145949774 EC50 = 1000 nM T58921 C04TKM 145949801 EC50 < 10 nM T58921 CLS49D 145950904 EC50 = 10 nM T58921 CT5BL8 145951025 EC50 = 94 nM T58921 CGE1B3 145951206 EC50 = 188 nM T58921 CQ6N2Z 145951479 EC50 = 62 nM T58921 CI08MP 145951689 EC50 = 335 nM T58921 C4GBZ5 145951912 EC50 < 10 nM T58921 CURD19 145952141 EC50 = 20 nM T58921 C9AST8 145952202 EC50 = 87 nM T58921 C8C2BN 145952574 EC50 = 356 nM T58921 C85OUK 145952859 EC50 = 129 nM T58921 CJA93S 145953039 EC50 = 23 nM T58921 C7EH8C 145953486 EC50 = 43 nM T58921 CQGS02 145953624 EC50 = 200 nM T58921 C96FER 145954306 EC50 = 1174 nM T58921 CV6L7A 145954353 EC50 = 118 nM T58921 CQ93BF 145954620 EC50 = 615 nM T58921 CT0HJ3 145955210 EC50 = 20 nM T58921 C0NLP6 145955315 EC50 = 474 nM T58921 CHW06J 145955457 EC50 = 318 nM T58921 CLW25D 145955603 EC50 = 736 nM T58921 CI4K0Z 145955653 EC50 = 40 nM T58921 CD3E4U 145955709 EC50 < 10 nM T58921 C5X9NS 145956690 EC50 = 1000 nM T58921 C8X9ZN 145956749 EC50 = 1895 nM T58921 C7URM5 145956965 EC50 = 230 nM T58921 CL0C9N 145956984 EC50 = 280 nM T58921 CS1W8N 145957036 EC50 = 25 nM T58921 C4C3IO 145957135 EC50 = 80 nM T58921 CJA0E5 145957371 EC50 = 20 nM T58921 CTIJ56 145957793 EC50 = 30 nM T58921 CCW82O 145958068 EC50 = 1000 nM T58921 CZ7X5B 145958164 EC50 < 10 nM T58921 CQ1X8H 145959158 EC50 = 391 nM T58921 CXR2V7 145959160 EC50 = 126 nM T58921 CA01SL 145959379 EC50 = 1132 nM T58921 CLW52V 145959485 EC50 = 65 nM T58921 C9VHW3 145959494 EC50 = 351 nM T58921 C08RPJ 145959499 EC50 = 30 nM T58921 CCR02D 145959510 EC50 = 50 nM T58921 CYVO42 145959628 EC50 = 395 nM T58921 CR54HC 145959653 EC50 = 200 nM T58921 CNH07S 145960072 EC50 = 717 nM T58921 C28YLS 145960168 EC50 = 269 nM T58921 CHL06X 145960211 EC50 = 101 nM T58921 CU14RO 145961656 EC50 = 4510 nM T58921 CFUV91 145962164 EC50 = 2320 nM T58921 CCF02H 145964530 IC50 = 6300 nM T58921 C56SHA 145964597 IC50 = 7600 nM T58921 C5DH4X 145964745 EC50 > 10000 nM T58921 C5H8EZ 145965425 IC50 = 6700 nM T58921 CT8AU9 145971273 EC50 = 746 nM T58921 CN01EU 145971719 EC50 = 1060 nM T58921 C9GPT8 145972429 EC50 = 1326 nM T58921 CA0RD6 145973168 EC50 = 71 nM T58921 C0LTV9 145973176 EC50 = 458 nM T58921 CJDH32 145975435 EC50 > 10000 nM T58921 C7J3IB 145976778 EC50 = 39670 nM T58921 C98CHS 145977976 IC50 = 7600 nM T58921 C0H2YI 145979664 EC50 = 140 nM T58921 C0KP3F 145980573 EC50 = 1750 nM T58921 C1Q6PV 145980608 EC50 = 2970 nM T58921 CY0AQ6 145981186 EC50 = 300 nM T58921 CKR43C 145981599 EC50 = 2030 nM T58921 C87UAM 145982210 EC50 = 4560 nM T58921 CFY8U2 145982433 EC50 = 1810 nM T58921 CW5YN6 145982467 EC50 = 33 nM T58921 C4D7TZ 145982651 EC50 > 10000 nM T58921 CT0YS3 145982746 EC50 > 10000 nM T58921 C65PGI 145982771 EC50 > 10000 nM T58921 CTFM01 145982798 EC50 > 10000 nM T58921 C65FME 145983252 EC50 > 10000 nM T58921 CH1XJ8 145983321 EC50 > 10000 nM T58921 C3WJZ8 145983637 EC50 > 10000 nM T58921 CP4W3R 145983705 EC50 > 10000 nM T58921 CT90OW 145983779 EC50 > 10000 nM T58921 CDZ5G0 145983839 EC50 = 22390 nM T58921 CFJ94I 145984084 EC50 > 10000 nM T58921 CH9MK6 145984248 EC50 = 25000 nM T58921 C8MUN3 145984355 EC50 = 8970 nM T58921 C8V7OD 145984577 EC50 > 10000 nM T58921 C4LN8E 145984731 EC50 > 10000 nM T58921 CIV2P1 145984795 EC50 > 10000 nM T58921 C0C2SU 145984820 EC50 > 10000 nM T58921 CQ1TB7 145984906 EC50 = 1690 nM T58921 CV84PQ 145985229 EC50 > 10000 nM T58921 CH9OI0 145985286 EC50 > 10000 nM T58921 CG8R3L 145985481 EC50 > 10000 nM T58921 C9LA1O 145985668 EC50 > 10000 nM T58921 CB47FE 145985838 EC50 = 9800 nM T58921 CRAK83 145985994 EC50 > 10000 nM T58921 CMAN27 145986012 EC50 = 18000 nM T58921 CA8JQ5 145986026 EC50 = 890 nM T58921 C9BR8T 145986189 EC50 = 15000 nM T58921 CAE95K 145986458 EC50 > 10000 nM T58921 CW7Y4G 145986696 EC50 = 1430 nM T58921 CBOR53 145986704 EC50 = 2020 nM T58921 C7V8GI 145987301 EC50 = 200 nM T58921 CVDF45 145987347 EC50 = 370 nM T58921 C0G2WE 145988431 EC50 = 1540 nM T58921 C75DSN 145989198 EC50 = 1750 nM T58921 CI39OJ 145989913 EC50 = 7750 nM T58921 CJ76KD 145990303 EC50 = 1850 nM T58921 C1CE8N 145991622 EC50 = 13 nM T58921 CV2FB6 145992078 EC50 = 1670 nM T58921 C4CJG3 145992093 EC50 = 197 nM T58921 C6F0LJ 145992170 EC50 = 1920 nM T58921 CP79UQ 145992176 EC50 = 2670 nM T58921 CL68BS 145992231 EC50 = 740 nM T58921 CI86HD 145992748 EC50 = 670 nM T58921 CCV39B 145994196 EC50 = 3170 nM T58921 CK5QF7 145994218 EC50 = 350 nM T58921 CFY20V 153392648 EC50 = 1140 nM T58921 CH7P2A 153392654 EC50 = 1320 nM T58921 CSN19A 153392659 EC50 = 590 nM T58921 C0D6EV 153392663 EC50 = 1390 nM T58921 C5A1NV 153392677 EC50 = 2550 nM T58921 C2TPX1 153392690 EC50 = 1480 nM T58921 C6HSO4 153392704 EC50 = 3390 nM T58921 C1BS3A 153392705 EC50 = 4250 nM T58921 C4F6XV 153392707 EC50 = 4210 nM T58921 CV14ZQ 153392749 EC50 = 1380 nM T58921 CI3LG0 153392752 EC50 = 1050 nM T58921 C47DGH 153392760 EC50 = 2410 nM T58921 CMG6B2 153392762 EC50 = 2620 nM T58921 CK0VH6 153392788 EC50 = 1750 nM T58921 C7X3AL 153763221 EC50 = 13200 nM T58921 CXN0T4 154649064 IC50 > 100000 nM T58921 CMG2U5 154649065 IC50 > 100000 nM T58921 C6JG4B 154649067 IC50 > 50000 nM T58921 CR6C2G 154649070 IC50 > 100000 nM T58921 C7DJ9Z 154649071 IC50 > 100000 nM T58921 CHYI48 154649073 IC50 = 78600 nM T58921 CB0WU5 155007664 IC50 > 50000 nM T58921 CPTL34 155491026 IC50 > 50000 nM T58921 C82EQJ 155510840 Ki = 13 nM T58921 C1R2HF 155510942 EC50 = 8660 nM T58921 CJ23ZU 155511506 IC50 = 8400 nM T58921 CD5QM6 155511861 EC50 = 457 nM T58921 C56XWT 155512000 IC50 > 50000 nM T58921 CSQ76T 155513005 IC50 = 15800 nM T58921 CY5X0R 155513188 IC50 = 3500 nM T58921 CKU7H8 155513886 Ki = 38 nM T58921 C3Z6VL 155514089 EC50 = 14000 nM T58921 CNKI04 155514770 IC50 = 5000 nM T58921 CWP3N5 155514845 IC50 = 13100 nM T58921 CICX19 155516325 EC50 = 1800 nM T58921 CB60UA 155516784 Ki = 52 nM T58921 C7ID2S 155517084 IC50 > 50000 nM T58921 C9NPC1 155517336 EC50 = 260 nM T58921 C1PUC8 155517399 EC50 = 3100 nM T58921 C2C4OZ 155518329 EC50 = 2800 nM T58921 C1POU5 155518522 EC50 = 4300 nM T58921 CLM6R2 155519632 IC50 = 6100 nM T58921 C6R1TF 155520683 EC50 = 6000 nM T58921 C59MDB 155521959 IC50 = 3900 nM T58921 CD2H3G 155522640 EC50 = 3310 nM T58921 CB65OD 155523050 EC50 = 2720 nM T58921 C9JL6O 155523070 IC50 > 50000 nM T58921 C2DO9Y 155523351 IC50 > 50000 nM T58921 C3GH8U 155523815 EC50 > 100000 nM T58921 CMC2S6 155523890 EC50 = 2194 nM T58921 CDS84A 155525533 IC50 > 50000 nM T58921 C95KYP 155526365 EC50 = 3100 nM T58921 C5BI8R 155527281 IC50 = 7200 nM T58921 CRL46F 155527309 EC50 = 991 nM T58921 C2LXU1 155527830 IC50 = 2600 nM T58921 CS3J1W 155527996 EC50 = 3700 nM T58921 CFYJ89 155529997 IC50 = 1900 nM T58921 C26IWH 155530219 EC50 = 2530 nM T58921 C9YTH8 155530420 EC50 = 770 nM T58921 C9D0QP 155531310 IC50 = 23900 nM T58921 C3Z5DW 155531660 EC50 = 1320 nM T58921 C6W2JV 155531862 EC50 > 100000 nM T58921 CZNI93 155531976 IC50 = 6400 nM T58921 C2O9VS 155532185 EC50 = 2.2 nM T58921 C21KSE 155532294 IC50 > 50000 nM T58921 CZ3JW4 155533609 IC50 = 3900 nM T58921 CO9YT5 155533758 EC50 > 100000 nM T58921 COG52I 155533929 Ki = 270 nM T58921 C4QF0W 155533937 EC50 = 1810 nM T58921 C63HSA 155534748 EC50 = 2939 nM T58921 CK89PE 155534755 EC50 = 2000000 nM T58921 CE7I8Q 155534885 EC50 = 33000 nM T58921 C0B5MT 155535253 EC50 = 160 nM T58921 CU1XD9 155535635 EC50 = 1230 nM T58921 CHC04X 155536991 EC50 = 50 nM T58921 CE2LR1 155538630 EC50 > 100000 nM T58921 C3KW1L 155538955 Ki = 144 nM T58921 COP7X8 155539171 IC50 > 10000 nM T58921 C3R9YL 155539254 EC50 = 28000 nM T58921 C0H4LN 155540058 IC50 = 6100 nM T58921 CJC0K1 155540534 EC50 = 1500 nM T58921 C83NUY 155541022 EC50 = 1360 nM T58921 C90LON 155541511 EC50 = 3.8 nM T58921 C7Q1FJ 155541575 IC50 > 50000 nM T58921 CSI9G7 155541727 EC50 = 4900 nM T58921 CJB39Q 155541750 EC50 = 1692 nM T58921 C5D3AP 155542482 EC50 = 460 nM T58921 CP4JL6 155544658 EC50 = 1000 nM T58921 CUJ1Z6 155544866 IC50 = 15100 nM T58921 CR36OJ 155545395 EC50 = 2360 nM T58921 C5Q6WG 155545482 EC50 = 2400 nM T58921 CA4RT6 155547357 IC50 = 11000 nM T58921 CG5ED6 155547434 IC50 = 9600 nM T58921 C0H7JO 155547646 EC50 = 1000 nM T58921 CL2QM6 155547835 EC50 = 2780 nM T58921 CSW56E 155548268 EC50 = 1500 nM T58921 CLS1M0 155549183 EC50 = 12100 nM T58921 C9X0CE 155549806 EC50 = 19 nM T58921 CDL1P9 155549826 IC50 = 4200 nM T58921 C87TQJ 155551096 EC50 = 3000 nM T58921 C9YTI8 155551777 EC50 = 730 nM T58921 C2MTF9 155552428 EC50 = 2900 nM T58921 CONR48 155553675 IC50 = 7500 nM T58921 C4BOE9 155554530 EC50 = 8670 nM T58921 CS7T3G 155554537 IC50 = 4700 nM T58921 CTYA23 155555023 IC50 = 9500 nM T58921 CV3RI5 155557021 Ki = 254 nM T58921 C0HRG6 155557561 Ki = 8 nM T58921 C52UDM 155557708 IC50 = 9400 nM T58921 CKXY48 155557717 Ki = 3799 nM T58921 CEI8F1 155558276 EC50 = 3700 nM T58921 CSN67H 155559112 IC50 = 2300 nM T58921 C9IXL2 155560109 IC50 = 3200 nM T58921 CBW05P 155560639 Ki = 27 nM T58921 CM52UW 155560868 EC50 = 2100 nM T58921 C4S9AD 155561084 IC50 > 50000 nM T58921 CF5IH8 155562394 EC50 = 5900 nM T58921 C3DN4K 155562634 EC50 = 700 nM T58921 C5GD4X 155563965 EC50 = 1090 nM T58921 C7WRN8 155564609 IC50 = 2500 nM T58921 C1KGW7 155565164 EC50 = 86 nM T58921 C5EUQ2 155565380 EC50 = 22 nM T58921 CD45PH 155565440 EC50 > 100000 nM T58921 CG02XL 155565451 EC50 > 10000 nM T58921 CU36GJ 155565702 IC50 = 5700 nM T58921 C3FK2M 155566781 EC50 = 1700 nM T58921 C47SHK 155566789 Ki = 38 nM T58921 CC63ZX 155568354 Ki = 13 nM T58921 C1I4MU 155568743 EC50 = 1060 nM T58921 CLS48D 155569070 Ki = 9461 nM T58921 CI24DH 155569680 EC50 = 84 nM T58921 D00ACX 644213 EC50 = 2 nM T58921 D00TFA 3392731 EC50 = 1100 nM T58921 D01POG 657048 EC50 = 243 nM T58921 D01RPM 11645581 IC50 = 980 nM T58921 D01UVA 181254 IC50 = 55000 nM T58921 D02TRN 445638 IC50 = 6400 nM T58921 D02TVS 985 IC50 = 30000 nM T58921 D02WFA 5281 IC50 = 30000 nM T58921 D03BPG 2777391 IC50 = 1000 nM T58921 D03LOG 5280450 IC50 = 6200 nM T58921 D04DYM 6518171 Ki = 0.0497 nM T58921 D04FVX 44220886 IC50 = 830 nM T58921 D05CLM 9870304 EC50 = 250 nM T58921 D06GYO 5282316 EC50 = 45 nM T58921 D06IHG 24836820 IC50 = 1610 nM T58921 D06MDX 11483970 EC50 = 480 nM T58921 D06NHI 9843045 Ki = 2.5 nM T58921 D06OBX 9975297 IC50 = 27000 nM T58921 D06RRD 2797 EC50 > 300000 nM T58921 D06TXM 24816385 EC50 = 3600 nM T58921 D06UVY 7019108 IC50 = 5200 nM T58921 D06VBQ 46233311 IC50 > 10000 nM T58921 D08OBF 11005 IC50 = 21000 nM T58921 D08QKF 9954280 IC50 = 26 nM T58921 D08QXD 9935197 EC50 = 23 nM T58921 D08UWZ 16725047 EC50 = 2400 nM T58921 D08ZYC 11595431 Ki < 3162.28 nM T58921 D09JII 9891946 EC50 = 5.2 nM T58921 D09XCX 5694 EC50 = 1600 nM T58921 D0A4EA 445639 IC50 = 4100 nM T58921 D0C5SV 5280934 IC50 = 6000 nM T58921 D0D0FQ 24762579 IC50 = 160 nM T58921 D0E7NO 2969 IC50 = 30000 nM T58921 D0F0MP 9889841 EC50 = 19 nM T58921 D0G9AI 25187914 IC50 = 18700 nM T58921 D0H4US 11149906 EC50 = 3600 nM T58921 D0HD9P 444899 IC50 = 1600 nM T58921 D0IW8V 7020170 IC50 = 18400 nM T58921 D0J3UU 11460087 EC50 = 2691.53 nM T58921 D0J9ZA 25185696 IC50 = 15100 nM T58921 D0K1TQ 9934458 EC50 = 2000 nM T58921 D0M7AT 25186251 IC50 = 15400 nM T58921 D0M9LL 44221100 IC50 = 39 nM T58921 D0N0UC 3893 IC50 = 30000 nM T58921 D0NM0G 2800647 IC50 > 10000 nM T58921 D0O2US 9870584 EC50 = 0.6166 nM T58921 D0P5QM 44221101 IC50 = 190 nM T58921 D0Q4EU 2286 IC50 = 100000 nM T58921 D0Q4UD 44220888 IC50 = 1680 nM T58921 D0R9VV 24180661 EC50 = 130 nM T58921 D0RL8P 24762580 EC50 = 160 nM T58921 D0T9ZL 2703 IC50 = 566 nM T58921 D0U5HX 24762578 EC50 = 260 nM T58921 D0W7RI 5311242 EC50 = 7910 nM T58921 D0W9WU 44220887 IC50 = 630 nM T58921 D0X3RZ 6997510 IC50 = 25800 nM T58921 D0X9UJ 44581800 IC50 = 820 nM T58921 D0XR8Q 1517 EC50 = 2500 nM T58921 D0YK9T 6603901 EC50 = 1824 nM T58921 D0Z4NW 44220889 IC50 = 1720 nM T58921 D0Z7OX 9890319 IC50 = 548 nM T40812 D01SHZ 9931954 IC50 = 0.5 nM T40812 D0GV8J 135565082 Ki = 0.85 nM T40812 D0J9HW 23725625 IC50 = 1 nM T40812 D00BMF 24958200 Ki = 4 nM T40812 D0F5TD 135565981 IC50 = 1 nM T40812 CXG7Y0 76959 IC50 = 77000 nM T40812 CJ2UB5 236501 IC50 > 100000 nM T40812 CYC75Z 622510 IC50 = 8300 nM T40812 C89WXS 2802462 IC50 = 34673.69 nM T40812 CR26SK 4163640 IC50 > 100000 nM T40812 CT9V6M 4826644 IC50 > 100000 nM T40812 C4P2UQ 8607850 IC50 > 100000 nM T40812 CGU16R 11842604 Ki = 2 nM T40812 CI0QP9 11960529 Ki = 5 nM T40812 CY1D6C 11960631 Ki = 2 nM T40812 CIL6Z8 11961092 Ki = 4 nM T40812 CG5A7W 16013152 IC50 > 19000 nM T40812 CBMF65 16013184 IC50 > 19000 nM T40812 C6V4TG 16013186 IC50 > 19000 nM T40812 C9LT3B 16031344 IC50 > 19000 nM T40812 CK6BD7 16665391 Ki = 1 nM T40812 COW9F1 16665466 Ki = 3 nM T40812 C5E2DM 16665467 Ki = 18 nM T40812 CR8FW9 16665469 Ki = 26 nM T40812 CAM95L 16665470 Ki = 3 nM T40812 C2E3GK 16665471 Ki = 23 nM T40812 C1I2OX 16665472 Ki = 10 nM T40812 CVP67B 16665552 Ki = 12 nM T40812 CV0W5R 16665702 Ki = 2 nM T40812 CB85MS 16665775 Ki = 18 nM T40812 C79ROY 16665776 Ki = 11 nM T40812 CYQ1W3 16665853 Ki = 3 nM T40812 CUS7D1 16666333 Ki = 1.5 nM T40812 CN4Y8E 18428049 Ki = 2 nM T40812 CZ6M5I 22431503 IC50 > 5011.87 nM T40812 CP9H4Y 22432631 IC50 > 5011.87 nM T40812 C1Y2MX 24772013 IC50 = 1 nM T40812 CL8Q0K 24772834 IC50 = 1 nM T40812 C96SVC 24852130 IC50 = 17 nM T40812 C5WQE0 24852132 IC50 = 32 nM T40812 C0IOR9 25015515 IC50 = 1000 nM T40812 CWIQ61 25190717 Ki = 11 nM T40812 C7UTZ4 25190739 Ki = 3 nM T40812 CS8KG2 25190740 Ki = 24 nM T40812 CPIK86 25190752 Ki = 2 nM T40812 CMXA39 28825277 IC50 > 100000 nM T40812 CSO1Z6 28825295 IC50 > 100000 nM T40812 CY5UH1 29717874 IC50 > 19000 nM T40812 CNI3Y5 44483163 IC50 > 18700 nM T40812 C1TPI7 44541920 Ki = 8 nM T40812 C8NH1A 44542066 Ki = 1 nM T40812 C3SOX5 44542366 Ki = 2 nM T40812 CBW72V 46173035 Ki = 4 nM T40812 CWF40I 56587957 IC50 > 100000 nM T40812 CD3HT9 67960134 IC50 > 100000 nM T40812 C7QLY3 71464718 IC50 > 10000 nM T40812 C6NUT0 71488522 IC50 = 1.9 nM T40812 C24XZF 71576800 IC50 > 10000 nM T40812 CI0GU8 71660496 IC50 > 170000 nM T40812 CZ1H8S 71681176 IC50 > 170000 nM T40812 C2RGP3 71681329 IC50 = 2200 nM T40812 CI5E8F 71681330 IC50 > 170000 nM T40812 CMC2J4 72193935 IC50 > 170000 nM T40812 C46DHU 72724967 IC50 > 170000 nM T40812 C5XHF0 72736758 IC50 = 0.22 nM T40812 CL3J2U 73056614 IC50 = 4700 nM T40812 CK67DZ 73293053 IC50 > 19000 nM T40812 CE4PM3 73293055 IC50 = 3800 nM T40812 CU3D9N 73388373 IC50 > 5011.87 nM T40812 CZY9U8 73441896 IC50 > 5011.87 nM T40812 C9VP6T 86276157 IC50 > 10000 nM T40812 C3XO5D 89649815 IC50 > 100000 nM T40812 C2XR5Q 92045137 IC50 = 1 nM T40812 CV0NZ7 105539834 IC50 > 100000 nM T40812 C02SDC 122423373 IC50 < 30 nM T40812 CV06MU 131801402 IC50 > 100000 nM T40812 C6PMI3 132576435 IC50 = 8.6 nM T40812 CGTF97 132576436 IC50 = 11.5 nM T40812 CLR6F7 132576437 IC50 = 4.1 nM T40812 C1OJM4 132576507 IC50 = 2.53 nM T40812 CRQ0L4 132576509 IC50 = 31.52 nM T40812 CMI36O 132601761 IC50 = 7.7 nM T40812 CMWX76 132601763 IC50 = 5.5 nM T40812 C34XLO 132601764 IC50 = 9.9 nM T40812 CV8MW6 132601765 IC50 = 7.2 nM T40812 CQ54WE 133053541 IC50 = 144 nM T40812 C9PI7O 135402338 IC50 = 2064 nM T40812 C0HQF2 135404247 IC50 = 2600 nM T40812 C47LAF 135418940 IC50 = 26.9 nM T40812 CIS9K5 135421564 IC50 > 100000 nM T40812 C4MW7F 135443732 IC50 = 1562 nM T40812 CZ9GA7 135449434 IC50 = 125 nM T40812 C8J2PC 135456762 IC50 = 3098 nM T40812 CHY9C3 135479130 IC50 = 4688 nM T40812 C7G6BQ 135513721 IC50 = 570 nM T40812 CDM28Q 135515514 IC50 = 500 nM T40812 CU3FW2 135566794 IC50 = 931 nM T40812 CG06FQ 135566852 IC50 > 19000 nM T40812 C8QDG3 135566882 IC50 = 2450 nM T40812 CNVM21 135566884 IC50 = 1760 nM T40812 C59OUK 135566970 IC50 > 10000 nM T40812 C7K5WL 135566971 IC50 > 10000 nM T40812 CU2I7X 135567125 IC50 = 6900 nM T40812 C37PTU 135567126 IC50 = 11481.54 nM T40812 C38XBR 135652704 IC50 = 2230 nM T40812 C4ZGO7 135741892 IC50 = 4080 nM T40812 CIL7K3 135742498 IC50 = 4.1 nM T40812 CS83CJ 135905416 IC50 = 990 nM T40812 CY94ZB 136215772 IC50 = 6350 nM T40812 C7JEG1 136215773 IC50 = 683 nM T40812 CF7O2U 136215774 IC50 > 100000 nM T40812 CFP0V5 136215897 IC50 = 10529 nM T40812 C19ELM 136219321 IC50 > 19000 nM T40812 C1VR8I 136219322 IC50 = 56400 nM T40812 CB19RP 136227775 IC50 = 6022 nM T40812 C8WOG5 136232687 IC50 > 19000 nM T40812 CR7Q4L 136232699 IC50 = 10400 nM T40812 C18MSY 136236981 IC50 = 1000 nM T40812 CW9H8J 136237302 IC50 = 3150 nM T40812 CV6OL8 136237316 IC50 = 32000 nM T40812 CA60VL 136237359 IC50 > 19000 nM T40812 C6JH2X 136237372 IC50 > 19000 nM T40812 C4DB3K 136237396 IC50 > 19000 nM T40812 CEWX52 136244045 IC50 > 19000 nM T40812 CR07BF 136244504 IC50 = 478.63 nM T40812 CUB67C 136404917 IC50 = 145 nM T40812 CF80AR 136491263 IC50 = 259 nM T40812 CYXU75 137348704 IC50 = 73 nM T40812 CW5ZQ2 137348705 IC50 = 124 nM T40812 CZXI62 137632887 IC50 = 1 nM T40812 CEP1D3 137633502 IC50 = 12.2 nM T40812 C0JBC6 137636342 IC50 > 100 nM T40812 CBV7D0 137636391 IC50 = 3.6 nM T40812 CW2M0P 137636515 IC50 > 100 nM T40812 CS7ZQ8 137637696 IC50 = 141 nM T40812 C0SQ6X 137638776 IC50 = 75 nM T40812 CPLK81 137639614 IC50 = 4.5 nM T40812 C71UPO 137640297 IC50 > 100 nM T40812 C9N2TJ 137642258 IC50 = 68 nM T40812 CD1O9L 137642588 IC50 > 100 nM T40812 C03XFD 137645265 IC50 = 38 nM T40812 CR2U1A 137645856 IC50 = 220 nM T40812 CY93WQ 137646242 IC50 = 9.1 nM T40812 C6P8EW 137646632 IC50 = 24 nM T40812 CT6DM0 137646713 IC50 = 5.8 nM T40812 CW9E5P 137647708 IC50 = 80 nM T40812 CF0ZT5 137648174 IC50 = 2.9 nM T40812 CT04QR 137648314 IC50 = 130 nM T40812 CFPV98 137650613 IC50 = 73 nM T40812 CM4X9L 137650820 IC50 > 100 nM T40812 CRV60J 137651431 IC50 = 74 nM T40812 C6USY9 137651641 IC50 = 19 nM T40812 CW5E8U 137651914 IC50 = 91 nM T40812 CH0TI5 137652048 IC50 = 49.12 nM T40812 C49QJY 137652661 IC50 = 11.9 nM T40812 C2N0KD 137654171 IC50 = 48 nM T40812 C1HE8S 137654622 IC50 = 5.02 nM T40812 CGXT37 137654655 IC50 > 100 nM T40812 CC4ON1 137656059 IC50 = 5.4 nM T40812 C24ROM 137657941 IC50 > 100 nM T40812 C8ABS0 137658730 IC50 > 100 nM T40812 CFVN90 137658777 IC50 = 34 nM T40812 C7B9ZV 137660079 IC50 = 40 nM T40812 CAH6B8 137660345 IC50 > 100 nM T40812 CS7LW6 137661452 IC50 = 100 nM T40812 C4R7VI 137701512 IC50 = 2717 nM T40812 C1XSH7 138594194 IC50 = 1240 nM T40812 CJW84M 138857416 IC50 = 10 nM T40812 C0QEY5 138857417 IC50 = 1.9 nM T40812 CWT79B 141466120 IC50 = 281 nM T40812 CW60NV 141466122 IC50 = 113 nM T40812 C6RZY8 141466124 IC50 = 117 nM T40812 C84QGZ 141466125 IC50 = 348 nM T40812 CZ2HI3 141466137 IC50 = 328 nM T40812 CV6BY1 141466145 IC50 = 359 nM T40812 C15IXJ 141466149 IC50 = 30 nM T40812 C64AQL 141466151 IC50 = 239 nM T40812 CVS5D0 141466159 IC50 = 86 nM T40812 CQ2S3B 141466167 IC50 = 109 nM T40812 CNTJ87 141466171 IC50 = 247 nM T40812 C1HKF6 141466173 IC50 = 87 nM T40812 CGI3Y5 141466177 IC50 = 42 nM T40812 C2TG0A 141466191 IC50 = 14 nM T40812 C6NM4Q 141466199 IC50 = 64 nM T40812 CXN16I 141466203 IC50 = 131 nM T40812 CBQ94P 141466205 IC50 = 219 nM T40812 C3YQJ1 141466206 IC50 = 196 nM T40812 CR2QP0 141466210 IC50 = 53 nM T40812 C53IRC 141466213 IC50 = 145 nM T40812 CR7WQ2 141466219 IC50 = 382 nM T40812 CN6M5U 141466229 IC50 = 324 nM T40812 CP1NZ6 141466233 IC50 = 140 nM T40812 C7E8DR 141466238 IC50 = 83 nM T40812 CX7PZ5 141639950 IC50 > 100000 nM T40812 CI09BF 141726120 IC50 = 67.8 nM T40812 CDTA25 145980841 IC50 = 99 nM T40812 C19UOE 145981852 IC50 = 356 nM T40812 C6VLE2 145987066 IC50 = 49 nM T40812 C2JN9I 145991734 IC50 = 149 nM T40812 CF01EN 145992009 IC50 = 70 nM T40812 C6RPG0 146014481 IC50 = 3.631 nM T40812 CLKO63 155510989 IC50 = 4.6 nM T40812 CKIA71 155512592 IC50 < 50 nM T40812 C70LFT 155512744 IC50 > 10 nM T40812 CA3OQ8 155514140 IC50 < 50 nM T40812 C57EUG 155517403 IC50 < 50 nM T40812 CSR58J 155518352 IC50 = 3 nM T40812 CI5KF8 155518636 IC50 = 4.786 nM T40812 CQ8IY2 155521429 IC50 > 10 nM T40812 CUI64O 155522393 IC50 = 3.467 nM T40812 CWK3O5 155524058 IC50 = 2.042 nM T40812 CN4EV1 155526203 IC50 < 50 nM T40812 CV5D1R 155526501 IC50 < 10 nM T40812 CLR5E0 155529239 IC50 < 50 nM T40812 CJ8H2Z 155530382 IC50 > 50 nM T40812 C2IL8E 155533692 IC50 = 3.802 nM T40812 CCS7P2 155534031 IC50 < 10 nM T40812 CCR95S 155534656 IC50 > 10 nM T40812 CS0O1N 155535359 IC50 > 10 nM T40812 CY8RJ7 155537249 IC50 = 3.981 nM T40812 C0ESO2 155537391 IC50 > 10 nM T40812 CR3B1W 155538039 IC50 < 50 nM T40812 C7W1DJ 155541447 IC50 = 1.585 nM T40812 CYWG48 155541643 IC50 = 1.585 nM T40812 CG0J7F 155545779 IC50 = 0.6457 nM T40812 C8FWY4 155549045 IC50 > 10 nM T40812 CBR3M2 155549878 IC50 < 50 nM T40812 C9B0VO 155549990 IC50 = 3.631 nM T40812 C6H3MX 155551959 IC50 > 10 nM T40812 CY1WI2 155552891 IC50 > 10 nM T40812 CJ8XG3 155553738 IC50 > 10 nM T40812 C0CGI2 155554382 IC50 < 50 nM T40812 CM48BL 155560098 IC50 < 50 nM T40812 C2A0TH 155560210 IC50 = 11.33 nM T40812 C0EC4U 155561767 IC50 > 10 nM T40812 CVX7E6 155562207 IC50 > 10 nM T40812 C6G1SQ 155562883 IC50 < 10 nM T40812 CZK5Q4 155566057 IC50 < 50 nM T40812 CJH14L 155566731 IC50 = 3.3 nM T40812 CTW09V 155568616 IC50 < 50 nM T40812 D03BQJ 688829 IC50 = 27542.29 nM T40812 D04WDX 4858 IC50 = 33.5 nM T40812 D06NKJ 135439437 IC50 = 1539 nM T40812 D0M9TW 25218518 IC50 = 8 nM T40812 D0OF1I 135417274 IC50 = 928 nM T40812 D0VY5O 9925908 Ki = 5 nM T15068 D07POC 176870 IC50 = 7400 nM T15068 D0AF6O 71731823 IC50 = 17 nM T15068 D0E6XR 3062316 IC50 > 50000 nM T15068 D0K8KX 5280343 IC50 = 1200 nM T15068 D0OB0F 5328940 IC50 = 538 nM T15068 D0R0MW 5329102 IC50 = 1600 nM T15068 D01SJT 11713159 IC50 = 1 nM T15068 D02UFQ 11620908 IC50 > 10000 nM T15068 D03HUX 49792852 IC50 > 10000 nM T15068 D03LWG 53235510 IC50 > 10000 nM T15068 D07EHV 44814409 IC50 > 10000 nM T15068 D0A6VD 25073775 IC50 = 1.5 nM T15068 D0E3TC 44259 EC50 = 11.32 ug.mL-1 T15068 D0N6NM 71721648 IC50 = 80 nM T15068 D0O0LS 25141092 IC50 = 140 nM T15068 D0Q7RE 16007391 Ki > 10000 nM T15068 D0S5RC 3025986 IC50 > 40000 nM T15068 D0S7HM 16041424 IC50 = 55 nM T15068 D0V6EV 25117126 IC50 = 0.6 nM T15068 D03BNU 59604787 IC50 > 3500 nM T15068 D0LF0O 135441202 IC50 = 165 nM T15068 D04FHB 6918852 Ki > 5000 nM T15068 D0T3ME 156422 IC50 = 2000 nM T15068 C63WLY 89644 IC50 = 1.5 ug.mL-1 T15068 C5JE2Z 104860 IC50 = 7.3 ug.mL-1 T15068 CI1NA5 159926 IC50 > 10 ug.mL-1 T15068 CYBA43 177458 IC50 > 10 ug.mL-1 T15068 CN05AH 406563 IC50 > 10000 nM T15068 CG2T7U 1290676 IC50 = 14640 nM T15068 CMKE97 3071991 IC50 = 156000 nM T15068 CCN9D5 3142817 IC50 = 900 nM T15068 CDG43V 3773533 IC50 = 3200 nM T15068 C26VMO 4366078 IC50 = 5700 nM T15068 C8IAR2 5281657 IC50 > 100000 nM T15068 CI68PW 5283685 IC50 = 9630 nM T15068 CXK0S6 5283727 IC50 = 13200 nM T15068 CDQ3M7 5359485 IC50 = 2.4 ug.mL-1 T15068 C54BYP 5360741 IC50 = 8.9 ug.mL-1 T15068 C4G9WR 9547398 IC50 > 100000 nM T15068 C76CUP 9547698 IC50 = 9920 nM T15068 COR9M1 9583941 IC50 = 11980 nM T15068 C12PKF 9871380 IC50 > 25000 nM T15068 CYW49X 9927718 IC50 > 25000 nM T15068 CN0AJ9 9934347 IC50 = 5.5 nM T15068 C4ER2C 10000911 IC50 = 160 nM T15068 CR8DA1 10024683 IC50 > 100000 nM T15068 CLA93G 10047202 IC50 = 10700 nM T15068 C3LCH5 10047545 IC50 > 100000 nM T15068 C7SFI1 10296883 IC50 = 8300 nM T15068 C4CP7K 10423452 IC50 = 15200 nM T15068 C83QWV 10714343 IC50 = 4560 nM T15068 C98XPQ 11152013 IC50 = 300 nM T15068 CZHR06 11154615 IC50 = 600 nM T15068 CEFH05 11175333 IC50 = 400 nM T15068 C0A5HJ 11185701 IC50 = 700 nM T15068 CH9Q6F 11186576 IC50 > 10000 nM T15068 C5V7YM 11200156 IC50 > 10000 nM T15068 C2GDX1 11203157 IC50 = 236 nM T15068 CT7I9X 11209256 IC50 = 900 nM T15068 C8G5WP 11210533 IC50 = 800 nM T15068 CI8J7Y 11214263 IC50 = 63 nM T15068 CBHV78 11221981 IC50 > 10000 nM T15068 C5WF9E 11222699 IC50 = 100 nM T15068 CZ0P9V 11224324 IC50 > 10000 nM T15068 CS8XT4 11224674 IC50 = 35 nM T15068 CZH6B3 11225226 IC50 = 119 nM T15068 CK2X8C 11232808 IC50 > 10000 nM T15068 CFN5T8 11257798 IC50 = 221 nM T15068 CFJO27 11270120 IC50 > 10000 nM T15068 CC2UM1 11270272 IC50 = 8000 nM T15068 C2DN0U 11278547 IC50 = 700 nM T15068 C2Y9WA 11278548 IC50 = 600 nM T15068 CP12JW 11293706 IC50 = 115 nM T15068 CW0J2R 11313605 IC50 = 2000 nM T15068 CQG2E7 11327482 IC50 = 63 nM T15068 CJ7HD6 11338577 IC50 = 126 nM T15068 C56EUK 11350824 IC50 = 3000 nM T15068 C4B7YV 11352629 IC50 = 298 nM T15068 CN4ZO5 11358569 IC50 > 10000 nM T15068 CBGM83 11362151 IC50 = 38 nM T15068 CZGC94 11363473 IC50 = 117 nM T15068 CT2LF4 11371398 IC50 > 10000 nM T15068 CXOI67 11374936 IC50 = 5060 nM T15068 C2WJV1 11392449 IC50 = 500 nM T15068 C2T9KR 11397993 IC50 = 54 nM T15068 CC48AW 11405903 IC50 = 1500 nM T15068 CZ3U0F 11419098 IC50 = 342 nM T15068 C63KST 11438633 IC50 = 700 nM T15068 CO1EP9 11443236 IC50 = 38 nM T15068 COVC47 11443737 IC50 = 73 nM T15068 CS39BT 11450357 IC50 = 200 nM T15068 C1D3ZI 11453158 IC50 = 93 nM T15068 C1VK8X 11460923 IC50 = 1200 nM T15068 CH45DI 11461644 IC50 > 10000 nM T15068 C6RJ9A 11465388 IC50 = 29 nM T15068 CEP4N0 11474859 IC50 > 10000 nM T15068 CGK4H5 11485032 IC50 = 7000 nM T15068 C7FT8B 11502189 IC50 = 34 nM T15068 CB9AC1 11525210 IC50 = 4 nM T15068 CL7X4Q 11530963 IC50 = 650 nM T15068 CPW07M 11545582 IC50 = 2810 nM T15068 CACS26 11561968 Ki > 10000 nM T15068 CO9KP5 11583459 IC50 > 10000 nM T15068 CN50CR 11596788 IC50 = 38 nM T15068 C5NB3M 11598628 IC50 = 1 nM T15068 CSM62L 11626920 IC50 = 478 nM T15068 C4FS2W 11669227 IC50 = 314 nM T15068 CU0E8O 11690457 Ki > 10000 nM T15068 CB0AP2 11705863 Ki > 10000 nM T15068 CE93KD 11771066 IC50 > 10000 nM T15068 C0MIE5 11773396 IC50 > 10000 nM T15068 C5AYN3 11774870 IC50 = 37 nM T15068 CCYB86 11948631 IC50 = 100 nM T15068 CASK85 11957393 IC50 = 200 nM T15068 C52GLP 11963310 IC50 > 125000 nM T15068 C5MI4N 14246200 IC50 = 11500 nM T15068 CDGF78 15282555 IC50 = 2100 nM T15068 C08NEU 15945881 IC50 = 266 nM T15068 C7LB4I 15949613 IC50 = 2600 nM T15068 CW0S4T 16118986 IC50 = 1.5 nM T15068 C5VPH9 16129448 IC50 = 136 nM T15068 C9IW5S 16730105 IC50 = 640 nM T15068 C9MNP2 17549086 IC50 > 50000 nM T15068 CYE2X8 19550325 IC50 = 1800 nM T15068 CEXI49 19550327 IC50 = 3200 nM T15068 C21OUW 21952403 IC50 = 9 nM T15068 C23ZPO 21952457 IC50 = 19 nM T15068 CS8D4H 21952489 IC50 = 1.9 nM T15068 C1TG0N 21952498 IC50 = 59 nM T15068 CA3I4T 24753787 IC50 > 50000 nM T15068 CCPS81 24764502 IC50 > 35000 nM T15068 C4V9GH 24894117 IC50 = 9500 nM T15068 CJH19T 24894883 IC50 = 50000 nM T15068 CKBY19 24894887 IC50 = 35000 nM T15068 C57BHF 24894888 IC50 = 28000 nM T15068 CB5TP8 24894992 IC50 = 28000 nM T15068 C32SUJ 24894993 IC50 = 40000 nM T15068 C41SIT 24894996 IC50 = 27000 nM T15068 CFW40U 24894997 IC50 = 43000 nM T15068 CN13JF 24899915 IC50 = 2.1 ug.mL-1 T15068 CBWR97 24899916 IC50 = 4.9 ug.mL-1 T15068 C9F2JD 24899917 IC50 > 10 ug.mL-1 T15068 C64MTI 24900160 IC50 > 10 ug.mL-1 T15068 CO2I6Q 24900161 IC50 > 10 ug.mL-1 T15068 CBK82P 25011729 IC50 = 19700 nM T15068 C0B7RT 25057409 IC50 > 10000 nM T15068 CTV54O 25123227 IC50 > 10000 nM T15068 CIG4H0 25178539 IC50 = 4400 nM T15068 C64KQP 25203958 IC50 > 10000 nM T15068 CFMU29 25229638 IC50 > 650 nM T15068 CKN0O6 25920890 IC50 = 3800 nM T15068 C2SM3W 42598243 IC50 = 17400 nM T15068 CJ5U1X 42639664 IC50 = 5.5 ug.mL-1 T15068 CEL61X 44229839 IC50 > 10000 nM T15068 CU4S0E 44410006 IC50 = 100 nM T15068 CBD9K7 44410115 IC50 = 7900 nM T15068 CUNY16 44410116 IC50 > 10000 nM T15068 CFA35K 44410125 IC50 > 10000 nM T15068 CWQ29H 44410126 IC50 > 10000 nM T15068 CR9GJ8 44410132 IC50 = 200 nM T15068 CSQE21 44410141 IC50 = 300 nM T15068 C94PWD 44410144 IC50 > 10000 nM T15068 C6MQX4 44410145 IC50 = 800 nM T15068 CPT47W 44410148 IC50 = 800 nM T15068 CYL07V 44410156 IC50 = 7500 nM T15068 CUR97Y 44410180 IC50 > 10000 nM T15068 C6BEN2 44410187 IC50 > 10000 nM T15068 CBA40F 44410189 IC50 > 10000 nM T15068 C27AVX 44410197 IC50 = 1000 nM T15068 CF82VO 44410221 IC50 > 10000 nM T15068 CH5E8V 44410264 IC50 > 10000 nM T15068 CVO4A5 44410293 IC50 > 10000 nM T15068 C9OR4E 44410294 IC50 = 500 nM T15068 CRS60L 44410299 IC50 = 800 nM T15068 C3STP8 44410300 IC50 = 500 nM T15068 C38AYI 44410304 IC50 = 9000 nM T15068 C1PXQ2 44410306 IC50 = 200 nM T15068 CQ2Y3I 44410307 IC50 = 200 nM T15068 CP91OG 44410336 IC50 > 10000 nM T15068 C3LQ1Y 44410967 IC50 > 10000 nM T15068 CJ5T7L 44410971 IC50 > 10000 nM T15068 CJF3S8 44410976 IC50 > 10000 nM T15068 CV9A4X 44410977 IC50 = 2820 nM T15068 CL46ZS 44410979 IC50 > 10000 nM T15068 CNM6C7 44410982 IC50 = 983 nM T15068 C8I7HY 44410983 IC50 = 434 nM T15068 C6G4KO 44410984 IC50 = 2710 nM T15068 C2L3ZJ 44410985 IC50 = 635 nM T15068 CH6QV5 44410989 IC50 = 882 nM T15068 CZ2DL7 44410990 IC50 = 331 nM T15068 C1TWQ4 44410991 IC50 > 10000 nM T15068 CS54AY 44410992 IC50 > 10000 nM T15068 C5QG7R 44410995 IC50 = 345 nM T15068 CK1G4H 44411002 IC50 = 397 nM T15068 CH1AQ2 44411003 IC50 = 278 nM T15068 CW7GX6 44411006 IC50 > 10000 nM T15068 C4Z2ON 44411010 IC50 = 242 nM T15068 CQZ93I 44411015 IC50 = 504 nM T15068 C09SYG 44411063 IC50 = 507 nM T15068 CK82NF 44411123 IC50 = 544 nM T15068 CFC17N 44411132 IC50 > 10000 nM T15068 CC02BO 44411133 IC50 = 262 nM T15068 CW84ZT 44411272 IC50 = 2840 nM T15068 C7ED5G 44411273 IC50 = 365 nM T15068 CWD9J8 44411274 IC50 = 1530 nM T15068 CYC38T 44411276 IC50 = 322 nM T15068 C2FSQ3 44411277 IC50 = 421 nM T15068 CQ6M8I 44411280 IC50 = 4110 nM T15068 C0K1JZ 44411281 IC50 = 5800 nM T15068 CC72NW 44411283 IC50 = 727 nM T15068 COC9Z8 44411284 IC50 = 1330 nM T15068 CRK65F 44411285 IC50 = 339 nM T15068 CV7SW1 44411286 IC50 = 7550 nM T15068 CJ89FX 44411288 IC50 > 10000 nM T15068 C4S2MP 44411289 IC50 = 3500 nM T15068 CNW39V 44411292 IC50 = 182 nM T15068 C7KA8P 44411298 IC50 > 10000 nM T15068 CPGJ34 44411304 IC50 = 4050 nM T15068 CO26CD 44411305 IC50 = 727 nM T15068 CU2XA9 44411309 IC50 > 10000 nM T15068 CI7E5M 44411310 IC50 = 235 nM T15068 CVT2Z8 44411330 IC50 = 1810 nM T15068 CVWS54 44411373 IC50 = 1510 nM T15068 CZU89Q 44411383 IC50 = 3230 nM T15068 C7P1ET 44411384 IC50 = 6500 nM T15068 C6TVJ0 44411402 IC50 = 1507 nM T15068 CI9RP8 44411403 IC50 = 5120 nM T15068 CN03IP 44411411 IC50 = 232 nM T15068 CGT50S 44411412 IC50 = 7320 nM T15068 CA5SJ6 44411413 IC50 = 831 nM T15068 CD8XG3 44411423 IC50 = 634 nM T15068 C3VRO9 44557921 IC50 > 10000 nM T15068 CUR98X 44562852 IC50 = 623 nM T15068 C0P2TQ 44562903 IC50 = 16 nM T15068 CF5Z1T 44562904 IC50 > 10000 nM T15068 CEJ8Y3 44562905 IC50 = 2200 nM T15068 CB8W7D 44562906 IC50 = 77 nM T15068 CIQ36A 44562948 IC50 = 46 nM T15068 CBU64Q 44562949 IC50 = 190 nM T15068 CF7I1N 44562995 IC50 = 170 nM T15068 C4EP1W 44562996 IC50 = 300 nM T15068 C2U3YS 44563035 IC50 = 810 nM T15068 CBWH32 44563037 IC50 = 0.5 nM T15068 CQC28T 44563059 IC50 = 880 nM T15068 CV3JH2 44563060 IC50 = 3200 nM T15068 CZW0B1 44563061 IC50 = 1300 nM T15068 C1Q7WR 44563062 IC50 = 0.94 nM T15068 CRJ5G1 44563101 IC50 = 3300 nM T15068 C9UEZ5 44563102 IC50 = 4000 nM T15068 CW0KF5 44563103 IC50 = 72 nM T15068 CU76FQ 44563134 IC50 = 4100 nM T15068 CSK2T1 44563136 IC50 = 1 nM T15068 C6QT0J 44622837 IC50 = 17000 nM T15068 CU3RF1 45139989 IC50 > 10000 nM T15068 CQGZ06 45139991 IC50 > 10000 nM T15068 CL1Z7W 45274615 IC50 > 125000 nM T15068 C4AD7X 45274823 IC50 = 18000 nM T15068 CX5S8P 45274824 IC50 > 125000 nM T15068 C6C9WM 45274825 IC50 = 1800 nM T15068 CMS63Y 45274934 IC50 = 1300 nM T15068 CP5LH0 45274936 IC50 > 125000 nM T15068 CAG3R0 45275054 IC50 > 125000 nM T15068 CQU52A 45275055 IC50 > 125000 nM T15068 CXZ2S5 45275165 IC50 > 125000 nM T15068 CW08BK 45275166 IC50 > 125000 nM T15068 C43NVG 45275167 IC50 = 1800 nM T15068 C7ON5A 46233287 IC50 > 10000 nM T15068 CCK54P 46852509 IC50 > 10000 nM T15068 CC57FP 46852510 IC50 = 551 nM T15068 C31UXV 46852812 IC50 = 122 nM T15068 C92ESA 49821674 IC50 = 4.25 nM T15068 CF91RS 49843531 IC50 > 10000 nM T15068 CD2K4R 50908681 IC50 = 194000 nM T15068 C2Y6QS 50938552 IC50 > 10000 nM T15068 C9NYP4 51036677 IC50 > 10000 nM T15068 C4WRY3 51037112 IC50 > 10000 nM T15068 CRI28Z 51037948 IC50 > 10000 nM T15068 CEQN27 52936621 Ki > 1000 nM T15068 CM24LF 52938983 IC50 = 4.13 nM T15068 CNPM14 53341082 IC50 > 3000 nM T15068 C8NA4L 53384644 IC50 > 30000 nM T15068 CWAY25 54586353 IC50 = 2100 nM T15068 CKOB52 54754160 EC50 = 10.79 ug.mL-1 T15068 C8AB1J 54759606 Ki = 530 nM T15068 C9ZFS1 54764923 IC50 = 16900 nM T15068 C2N1XJ 56657923 EC50 = 12.15 ug.mL-1 T15068 C7RHL1 56657924 EC50 = 26.15 ug.mL-1 T15068 C3E8GJ 56657925 EC50 = 13.69 ug.mL-1 T15068 C46BUN 56661448 EC50 = 13.98 ug.mL-1 T15068 CN67IC 56664891 EC50 = 23.73 ug.mL-1 T15068 CTQS47 56668307 EC50 = 18.11 ug.mL-1 T15068 CEH31Y 56668417 IC50 = 17 nM T15068 C9T2BN 56675203 EC50 = 19.02 ug.mL-1 T15068 C53NYE 56679785 EC50 = 17.74 ug.mL-1 T15068 C6W0UF 56683115 EC50 = 21.04 ug.mL-1 T15068 CUT2G8 56835062 IC50 = 420 nM T15068 C5FY9U 56945728 IC50 = 21 nM T15068 CV6Z5P 56952427 IC50 = 17.1 nM T15068 CV0T6Y 56953221 IC50 = 31.9 nM T15068 CPHX64 57325478 IC50 > 50000 nM T15068 CQ9BW4 57325479 IC50 > 50000 nM T15068 C5USP1 57327769 IC50 = 420 nM T15068 CZYM98 57327842 IC50 = 920 nM T15068 CS49KB 57327913 IC50 = 960 nM T15068 C10WYL 57390861 IC50 = 205 nM T15068 C5O1HP 57392676 IC50 = 14 nM T15068 C6SKR3 57392677 IC50 = 167 nM T15068 C3J4NV 57394381 IC50 = 14 nM T15068 CK74ND 57394382 IC50 = 114 nM T15068 C43EQN 57394383 IC50 = 1010 nM T15068 C1V9MC 57394384 IC50 = 2040 nM T15068 CKS67A 57396146 IC50 = 660 nM T15068 CWJ70D 57397964 IC50 = 39 nM T15068 CAQ9D6 57397965 IC50 > 1000 nM T15068 CZX8R7 57399606 IC50 = 48 nM T15068 CL9Z2D 57401363 IC50 = 1340 nM T15068 C8F4ME 57401364 IC50 = 33 nM T15068 C9GN1M 57403118 IC50 = 55 nM T15068 C56CSP 57403119 IC50 = 1230 nM T15068 CVK0G4 58056356 IC50 > 50000 nM T15068 C47AGK 59284564 IC50 = 320 nM T15068 CT3EW2 59292007 IC50 > 1000 nM T15068 COH62U 60097413 IC50 > 10000 nM T15068 C1MR8Q 60097495 IC50 > 9000 nM T15068 C4SGZ6 60165992 IC50 = 92000 nM T15068 C98NOD 60165993 IC50 = 38000 nM T15068 C3WIX5 60165994 IC50 = 58000 nM T15068 C0G5WC 60165995 IC50 = 69000 nM T15068 CEQ07N 60166135 IC50 = 24000 nM T15068 CRV13A 60166136 IC50 > 100000 nM T15068 CLP62H 60166137 IC50 = 27000 nM T15068 C9X0ZC 60166139 IC50 = 5200 nM T15068 CWPZ07 60166141 IC50 = 3400 nM T15068 C37NKO 67129970 IC50 > 10000 nM T15068 CK80LJ 67130050 IC50 = 4790 nM T15068 CV63UL 67240318 IC50 > 10000 nM T15068 C7GRV2 68755406 IC50 > 10000 nM T15068 C3ETH7 70678491 IC50 = 4770 nM T15068 C7UYO2 70678492 IC50 = 7860 nM T15068 CAO2N0 70789288 IC50 = 500 nM T15068 C15TYU 71272361 IC50 = 45 nM T15068 C98MXV 71272465 IC50 = 177 nM T15068 CR5H0G 71277531 IC50 = 195 nM T15068 CE6DK5 71277533 IC50 > 10000 nM T15068 CL84RM 71277535 IC50 = 8900 nM T15068 CO08QB 71277539 IC50 = 220 nM T15068 C8B5IZ 71277542 IC50 = 2400 nM T15068 CE5AY6 71277544 IC50 = 8800 nM T15068 CV37JZ 71277560 IC50 > 10000 nM T15068 CB8HX7 71277567 IC50 = 51 nM T15068 CJS50G 71277569 IC50 = 4500 nM T15068 CF4PS5 71277570 IC50 = 170 nM T15068 CDP79T 71277572 IC50 = 37 nM T15068 C2NIW3 71277573 IC50 > 10000 nM T15068 CM09RU 71277577 IC50 = 45 nM T15068 CYE15N 71277578 IC50 = 130 nM T15068 CCX43N 71277591 IC50 > 10000 nM T15068 C8GIE2 71277641 IC50 > 10000 nM T15068 CW1P5B 71450692 IC50 = 608 nM T15068 C5Z6EG 71452514 IC50 > 10000 nM T15068 CEBO91 71452977 IC50 > 10000 nM T15068 CI03HX 71454272 IC50 > 10000 nM T15068 C0ML9S 71456031 IC50 = 473 nM T15068 CT8UI0 71457834 IC50 > 10000 nM T15068 CX54WG 71504922 IC50 = 910 nM T15068 CISP56 71504923 IC50 = 4800 nM T15068 C9E2SI 71504924 IC50 > 10000 nM T15068 C3GZV1 71505118 IC50 = 700 nM T15068 CSM8Q3 71524871 IC50 = 13600 nM T15068 CQ34CK 71524919 IC50 = 10300 nM T15068 CZQ2S4 71524965 IC50 = 28700 nM T15068 C8A9IN 71525006 IC50 = 9900 nM T15068 C0M4LC 71525009 IC50 = 6200 nM T15068 CCN01X 71547862 IC50 > 10000 nM T15068 CB3SO2 71567006 IC50 = 77 nM T15068 C3JNR4 71567007 IC50 = 3500 nM T15068 C0RJC8 71567008 IC50 = 990 nM T15068 CN9ML8 71567009 IC50 = 2400 nM T15068 CQJ06M 71567010 IC50 = 4300 nM T15068 CC6SH1 71567143 IC50 > 30000 nM T15068 C4TEY9 71567144 IC50 = 2000 nM T15068 CVH2S1 71567146 IC50 = 19000 nM T15068 C98HZS 71567147 IC50 = 1400 nM T15068 CQR8U1 71567148 IC50 > 30000 nM T15068 CDJY72 71568837 IC50 = 880 nM T15068 C8CAG7 71578921 IC50 = 3200 nM T15068 CVT67X 71608474 IC50 = 37 nM T15068 CY8VM4 71695585 IC50 = 7000 nM T15068 CW9U4T 71712420 IC50 = 1200 nM T15068 CW8R2M 71712555 IC50 = 9500 nM T15068 CU4Z5S 71712556 IC50 = 9800 nM T15068 CZ9S7R 71712557 IC50 = 12100 nM T15068 CJ4UG2 71712558 IC50 = 7100 nM T15068 C9UK4G 71712559 IC50 = 7600 nM T15068 CMP0L6 71712560 IC50 = 7100 nM T15068 CMVC79 71712561 IC50 = 8300 nM T15068 CSJ82Y 71712707 IC50 = 14200 nM T15068 C3FSK6 71712708 IC50 = 15800 nM T15068 CX2YL9 71712709 IC50 = 7500 nM T15068 CFAH06 71712710 IC50 = 7000 nM T15068 C04RLN 71712711 IC50 = 9100 nM T15068 C23YMQ 71712712 IC50 = 23700 nM T15068 CBTX24 71712713 IC50 = 33800 nM T15068 CA1Z4P 71712855 IC50 = 8600 nM T15068 C0I4KN 71712856 IC50 = 9200 nM T15068 C0HI4T 71712857 IC50 = 28500 nM T15068 CDQ9C7 71712858 IC50 = 33600 nM T15068 C5JB7Y 71717974 IC50 = 640 nM T15068 CK29UP 71719799 IC50 = 57 nM T15068 C3AGY0 71812600 IC50 = 5100 nM T15068 CBNV42 71812783 IC50 = 9200 nM T15068 CO8D9S 71812784 IC50 = 400 nM T15068 CLU3E2 71812785 IC50 = 2200 nM T15068 C84UWZ 71812786 IC50 = 6100 nM T15068 CZE23S 71812787 IC50 = 6000 nM T15068 CY9J8G 71812788 IC50 = 5200 nM T15068 CST1Y3 71812964 IC50 = 23800 nM T15068 CO7BL4 71812965 IC50 = 10200 nM T15068 C1SO7W 71812966 IC50 = 17900 nM T15068 CT5X4U 71812967 IC50 = 6100 nM T15068 C76KXR 71812968 IC50 = 1500 nM T15068 CJGA85 71812969 IC50 = 21100 nM T15068 CP6E7H 71813141 IC50 = 300 nM T15068 CZWV34 71813142 IC50 = 2300 nM T15068 CI9R5X 71813143 IC50 = 160 nM T15068 CBXJ06 71813144 IC50 = 440 nM T15068 CZ7IB0 71813145 IC50 = 1000 nM T15068 CL96SA 71813328 IC50 = 1900 nM T15068 C6Z1RW 71813329 IC50 = 65900 nM T15068 CM06VW 71813330 IC50 = 41300 nM T15068 CX61UD 71813331 IC50 = 7900 nM T15068 CSD6M7 71813332 IC50 = 50800 nM T15068 CLS6A0 71813493 IC50 = 35900 nM T15068 C7S8FO 71813494 IC50 = 54300 nM T15068 C1FB9X 71813495 IC50 = 125600 nM T15068 C2OV4Z 72189207 IC50 = 7700 nM T15068 CW4E9O 72189514 IC50 = 9100 nM T15068 CAVB46 72189515 IC50 > 10000 nM T15068 C4KUM3 72189516 IC50 > 10000 nM T15068 CR5Y6U 72189517 IC50 = 8400 nM T15068 C46FSX 72189518 IC50 > 10000 nM T15068 CBW0G9 72189519 IC50 > 10000 nM T15068 CC0DB5 72189807 IC50 > 10000 nM T15068 CUQ69N 72189808 IC50 > 10000 nM T15068 C1V7PU 72189809 IC50 > 10000 nM T15068 CC1SR3 72189810 IC50 > 10000 nM T15068 C9NCE7 72189811 IC50 = 5000 nM T15068 C2ZF9X 72190130 IC50 > 10000 nM T15068 CXH2S6 72190131 IC50 > 10000 nM T15068 C12KEZ 72190132 IC50 > 10000 nM T15068 CW64OR 72190133 IC50 > 10000 nM T15068 C01FBU 72547701 IC50 = 17380 nM T15068 CV4Y7A 72723312 IC50 = 10400 nM T15068 CQJ7X3 73349094 IC50 = 41900 nM T15068 C1ZD6C 73350669 IC50 = 57800 nM T15068 C3UC9H 73891099 IC50 = 420 nM T15068 C1GXB5 76309580 IC50 = 19380 nM T15068 CV8QX0 76310169 IC50 = 16300 nM T15068 CCQG84 76324167 IC50 = 9170 nM T15068 CA5L4W 76324771 IC50 = 20600 nM T15068 C9GO0P 76328313 IC50 = 7520 nM T15068 C39FTZ 76335685 IC50 = 7780 nM T15068 CQZ0L8 78158242 IC50 = 3.1 nM T15068 CJHE92 86233364 IC50 = 3800 nM T15068 CSH3G2 86287525 IC50 = 6900 nM T15068 C03NKD 90643488 IC50 = 6550 nM T15068 C3TI1B 90643489 IC50 = 3420 nM T15068 CK3W2E 90643490 IC50 = 18420 nM T15068 CJ7GT9 90643491 IC50 = 12430 nM T15068 CMN14F 90643492 IC50 = 10340 nM T15068 CDY54C 90643493 IC50 = 1750 nM T15068 CFO1Y9 90643494 IC50 = 4340 nM T15068 C9FSC3 90643495 IC50 = 5210 nM T15068 CAHP28 90643496 IC50 = 8010 nM T15068 CTAJ97 90643497 IC50 = 23540 nM T15068 C83KOD 90643498 IC50 = 16210 nM T15068 CDM9C4 90643499 IC50 = 26540 nM T15068 CG7YM5 90643500 IC50 = 30070 nM T15068 CP1E3A 90643501 IC50 = 24430 nM T15068 CPD4T3 90643502 IC50 = 28670 nM T15068 CM0OE7 90643503 IC50 = 450 nM T15068 C4KOQ3 90643504 IC50 = 1010 nM T15068 C2WAC8 90643505 IC50 = 20560 nM T15068 CY0UC4 90645194 IC50 > 10000 nM T15068 CBG6E7 91885506 IC50 = 1 nM T15068 C0Y8ZK 91933875 IC50 > 100 nM T15068 CH3TU5 101913593 IC50 = 330 nM T15068 CF72PB 101913594 IC50 = 230 nM T15068 C2Y1HS 101913596 IC50 = 120 nM T15068 C3N5IY 117955447 IC50 = 2.4 nM T15068 C5T4WU 117955577 IC50 = 2.2 nM T15068 C2T4MB 117955613 IC50 = 42 nM T15068 C07ACT 117955744 IC50 = 7 nM T15068 C5K2DA 117955863 IC50 = 4 nM T15068 C50ANY 117955890 IC50 = 9.3 nM T15068 CY7BI2 118706214 IC50 > 10000 nM T15068 C3KLI5 118723185 IC50 > 100000 nM T15068 C2FBJ1 118725339 IC50 = 280 nM T15068 C42DLU 118725340 IC50 = 570 nM T15068 C7LNE1 118725341 IC50 = 870 nM T15068 C30RQV 118725342 IC50 = 1200 nM T15068 CNJ9O6 118725429 IC50 = 310 nM T15068 CJC32Y 118725430 IC50 = 370 nM T15068 CPU83W 118725431 IC50 = 570 nM T15068 CZ4B8W 118725432 IC50 = 510 nM T15068 C5IV0R 118725433 IC50 = 710 nM T15068 CR7G8Y 118725434 IC50 = 1120 nM T15068 C47WPX 118725435 IC50 = 920 nM T15068 CI6A3Y 118725436 IC50 = 1730 nM T15068 CG23JF 118725437 IC50 = 500 nM T15068 CEM6S7 118725438 IC50 = 1050 nM T15068 C6XZ1P 118725439 IC50 = 50 nM T15068 CY5OJ7 118725440 IC50 = 880 nM T15068 C93QXF 118725441 IC50 = 240 nM T15068 CX4Y9U 118725442 IC50 = 280 nM T15068 CQ7NU0 118725443 IC50 = 220 nM T15068 C1T5KC 118725444 IC50 = 370 nM T15068 CLN9U2 118725445 IC50 = 180 nM T15068 C4QS6F 118725446 IC50 = 840 nM T15068 C14HRP 118725447 IC50 = 8910 nM T15068 CQCX41 118737057 IC50 > 10000 nM T15068 CG9Q1H 121320416 IC50 = 891 nM T15068 CLP1V0 127030406 IC50 = 1900 nM T15068 C0M4FL 127031111 IC50 = 3900 nM T15068 CUBC85 127031112 IC50 = 10630 nM T15068 C7M0KI 127031113 IC50 = 2600 nM T15068 C75GFW 127031114 IC50 = 2900 nM T15068 CGF5D4 127031425 IC50 = 3300 nM T15068 C3I2QA 127031426 IC50 = 1100 nM T15068 CVD9G8 127031942 IC50 = 2200 nM T15068 C7VD3N 127031993 IC50 = 250 nM T15068 C0RF2K 127031994 IC50 = 6600 nM T15068 CD9T5M 127031996 IC50 = 3900 nM T15068 C68BDG 127031997 IC50 = 3800 nM T15068 C43ZQY 127031998 IC50 = 3200 nM T15068 C45BMP 127032859 IC50 = 26500 nM T15068 C62MGZ 127033456 IC50 = 3500 nM T15068 CUO0C5 132156633 IC50 > 10000 nM T15068 C1FZ0K 132576331 IC50 = 82.5 nM T15068 CWT83G 132576332 IC50 = 84.7 nM T15068 C8W1JX 132576333 IC50 = 86.7 nM T15068 C54AQT 132576334 IC50 = 84.6 nM T15068 C9JBR2 132576335 IC50 = 108.8 nM T15068 CL6E4J 132601725 IC50 = 15600 nM T15068 C0YNT6 132942276 IC50 = 780 nM T15068 CMXH52 134130812 IC50 = 17 nM T15068 CMAJ86 134132390 IC50 = 11.4 nM T15068 CG9S2T 134132953 IC50 = 9.2 nM T15068 C3FXQ8 134133959 IC50 = 7496 nM T15068 CQ8SO0 134134585 IC50 = 8.6 nM T15068 CKGX09 134136179 IC50 = 0.51 nM T15068 CC82TI 134141407 IC50 = 177 nM T15068 CW04KZ 134141466 IC50 = 3.8 nM T15068 C7QNE8 134143033 IC50 = 27 nM T15068 C5WE2S 134147409 IC50 = 1.26 nM T15068 CFG60Q 134148895 IC50 = 8.5 nM T15068 CV02ZU 134149369 IC50 = 3.3 nM T15068 C6XHZ0 134149712 IC50 = 21 nM T15068 C04SWY 134150465 IC50 = 0.51 nM T15068 CZBC58 134153003 IC50 = 14 nM T15068 CJ47PZ 134153599 IC50 = 5.75 nM T15068 C73UZY 134155285 IC50 = 10.2 nM T15068 C1IQ6Y 134155909 IC50 = 3.2 nM T15068 CP9MH0 134156043 IC50 = 4.34 nM T15068 C2UJ9A 134156448 IC50 = 3.21 nM T15068 C7H8GQ 134157229 IC50 = 6.5 nM T15068 C29PWN 135886762 IC50 > 50000 nM T15068 C9W6BT 136002660 IC50 = 1200 nM T15068 CD9CT6 136002661 IC50 = 150 nM T15068 C4T9KZ 136002662 IC50 = 180 nM T15068 CHA4N2 136013680 IC50 > 10 nM T15068 C48DLS 136123445 IC50 = 94 nM T15068 CZ7EX0 136183413 IC50 = 5490 nM T15068 C6HW4E 136206295 IC50 = 11400 nM T15068 CU9P3M 136206296 IC50 = 10400 nM T15068 C1YUD0 136219394 IC50 > 10 nM T15068 C2FS9X 136240066 IC50 = 2410 nM T15068 CIU8W3 136254389 IC50 > 10 nM T15068 CXC69T 137321158 IC50 = 89 nM T15068 C4H9RG 137633210 IC50 = 110 nM T15068 CQ7T3G 137633302 IC50 = 2450 nM T15068 C5Z6EY 137633434 IC50 = 1120 nM T15068 CXE91W 137633895 IC50 = 340 nM T15068 CI1E8V 137634241 IC50 = 5500 nM T15068 CVD9E7 137636479 IC50 = 2400 nM T15068 CT91WL 137636559 IC50 = 2500 nM T15068 CRD5K6 137637150 IC50 = 1900 nM T15068 CVKM05 137639598 IC50 = 235.9 nM T15068 C0M2DV 137642413 IC50 = 7800 nM T15068 CZDI94 137645280 IC50 = 9500 nM T15068 CW5N0Q 137645598 IC50 = 3500 nM T15068 CTRW26 137645712 IC50 = 640 nM T15068 C50ISY 137647338 IC50 = 1970 nM T15068 CR02UC 137649431 IC50 = 2450 nM T15068 C3XQ4T 137649572 IC50 = 2900 nM T15068 CX9BD8 137651363 IC50 = 2000 nM T15068 CNM9Q4 137652602 IC50 = 2760 nM T15068 C7Z3OK 137652842 IC50 = 5500 nM T15068 C4Q0FZ 137652901 IC50 = 1460 nM T15068 CNB10S 137653041 IC50 = 1800 nM T15068 CB7QK0 137654886 IC50 = 2450 nM T15068 CC9T6P 137655041 IC50 = 1160 nM T15068 CA8KV2 137655141 IC50 = 870 nM T15068 C5C1FY 137655236 IC50 = 3120 nM T15068 C3HOL2 137655244 IC50 = 113.8 nM T15068 C4U6BC 137657356 IC50 = 1200 nM T15068 CJF6G7 137659313 IC50 = 7000 nM T15068 C36AXC 137660619 IC50 = 230 nM T15068 C8PJ4E 137661142 IC50 = 560 nM T15068 C5I8WZ 137661276 IC50 = 109.2 nM T15068 C0Y4XD 137662183 IC50 = 1000 nM T15068 C1UGS8 138454773 IC50 = 6.5 nM T15068 C8WE0V 138454785 IC50 = 25 nM T15068 CLHF74 138454791 IC50 = 0.07 nM T15068 CP5B7J 145964501 IC50 = 10.69 nM T15068 C9E1KF 145965257 IC50 = 5.69 nM T15068 C40OXF 145969869 IC50 = 6.18 nM T15068 CE2CZ0 145971411 IC50 = 4.65 nM T15068 CCM36L 145977422 IC50 = 5.01 nM T15068 C09CIA 146309709 IC50 = 14.5 nM T15068 CS8DW7 146309712 IC50 = 11.3 nM T15068 CFDQ64 146309714 IC50 = 14.7 nM T15068 CU8EJ7 146309721 IC50 = 4.7 nM T15068 CN8JR0 146309723 IC50 = 12.7 nM T15068 CU19YP 146309726 IC50 = 9.7 nM T15068 C5QVW7 146314935 IC50 = 10.7 nM T15068 CJ3VM4 147665857 IC50 = 175.4 nM T15068 C0J6TU 148252562 IC50 = 316.3 nM T15068 CW4QJ0 155512932 IC50 = 32.7 nM T15068 C2MD1Q 155513187 IC50 > 10000 nM T15068 CFN2T7 155517127 IC50 = 38 nM T15068 CR8H5N 155517701 IC50 = 91.8 nM T15068 CY9MH3 155517945 IC50 = 17.2 nM T15068 C86HPW 155518524 IC50 > 100000 nM T15068 CWK25Y 155518971 IC50 = 156.1 nM T15068 CW0ML1 155519156 IC50 = 150.8 nM T15068 C83SFL 155519688 IC50 = 126.4 nM T15068 C9T2BE 155520510 IC50 = 5.4 nM T15068 C3KSO9 155521946 IC50 = 176.6 nM T15068 C7SQJ4 155522728 IC50 = 6.8 nM T15068 C9I8TL 155523032 IC50 = 75.8 nM T15068 CI92YO 155523359 IC50 = 154.2 nM T15068 CX7M8L 155523717 IC50 = 14 nM T15068 CC1E0N 155524460 IC50 = 51.1 nM T15068 CZ68NO 155525555 IC50 = 10.3 nM T15068 C8JAQ7 155528659 IC50 = 25.6 nM T15068 CT0M7R 155528770 IC50 = 23 nM T15068 CP2AC5 155531043 IC50 = 347.5 nM T15068 CS41DB 155531735 IC50 = 21.1 nM T15068 C0SZY8 155532110 IC50 = 15.5 nM T15068 CO78TC 155533170 IC50 = 26.2 nM T15068 CG8V7O 155533749 IC50 = 8.57 nM T15068 CI5N1K 155534857 IC50 = 64.1 nM T15068 CTDO67 155535237 IC50 = 2.58 nM T15068 CJ2NP6 155535716 IC50 = 16.7 nM T15068 C78MZC 155536330 IC50 = 18 nM T15068 C6RT0B 155538008 IC50 = 5.1 nM T15068 C3OF6I 155538017 IC50 = 38.7 nM T15068 CTSM92 155538441 IC50 = 11 nM T15068 C5U8YA 155539566 IC50 = 9.3 nM T15068 C6MF1J 155539907 IC50 = 185.6 nM T15068 C84BMY 155540664 IC50 = 20.6 nM T15068 C3I2UE 155541058 IC50 = 62.1 nM T15068 CQ2HO5 155545546 IC50 = 23.1 nM T15068 C8T6AI 155549540 IC50 = 21.9 nM T15068 CO1V2N 155550374 IC50 = 34.5 nM T15068 CQM0B1 155550672 IC50 = 85 nM T15068 CJY2N4 155552497 IC50 = 5.8 nM T15068 C3K4BL 155555187 IC50 = 9.4 nM T15068 CBDZ80 155561484 IC50 = 7.28 nM T15068 C2BYX4 155561587 IC50 = 64.4 nM T15068 CW7S9H 155563239 IC50 = 9.1 nM T15068 C9RMB0 155564807 IC50 = 132.6 nM T15068 CMXF91 155566714 IC50 = 5.17 nM T15068 CHPT86 155567813 IC50 = 38.2 nM T15068 C10EFN 155568019 IC50 = 506.7 nM T15068 C9ZLX1 155568781 IC50 = 80.8 nM T15068 CO67YZ 155569323 IC50 = 82 nM T15068 D02QAZ 11612883 IC50 = 50 nM T15068 D06HVH 54613583 IC50 > 10000 nM T15068 D06LJL 9916282 IC50 = 4000 nM T15068 D06QWO 14824655 IC50 > 10 ug.mL-1 T15068 D08HFG 24809764 IC50 > 10000 nM T15068 D09HVH 135566652 IC50 > 10 nM T15068 D09PTP 57325421 IC50 = 25 nM T15068 D0A1CM 5281855 IC50 = 3110 nM T15068 D0AY0F 70698427 IC50 = 2200 nM T15068 D0E7VO 59627005 IC50 = 17.2 nM T15068 D0G3SZ 6918469 IC50 > 10 ug.mL-1 T15068 D0J3LR 11634725 Ki > 10000 nM T15068 D0K5UF 72710568 IC50 = 16 nM T15068 D0M4SY 135440466 IC50 = 150 nM T15068 D0YZ7H 9797370 IC50 > 100000 nM T42724 D09GOS 2812 IC50 = 70 nM T42724 D00BUR 216327 IC50 = 12 nM T42724 CK4L6D 68992 IC50 > 10000 nM T42724 CL9WP7 3657291 IC50 = 3150 nM T42724 CF38UJ 4419328 IC50 = 550 nM T42724 C32FGI 4447360 IC50 = 1750 nM T42724 C6F5HV 9967816 IC50 = 15 nM T42724 C1LB2Z 20684854 IC50 = 15 nM T42724 C4OF9S 21705158 IC50 = 17 nM T42724 C9PC8V 44592758 IC50 = 1400 nM T42724 CN1PC9 44592783 IC50 = 2400 nM T42724 C3ESW7 44592784 IC50 = 16000 nM T42724 C46XRM 44592785 IC50 = 1300 nM T42724 CZY20B 71520370 IC50 = 7800 nM T42724 C0T9BG 71520371 IC50 > 33000 nM T42724 C4OBM9 71520373 IC50 = 10000 nM T42724 CXT3L0 71520486 IC50 = 31000 nM T42724 CA3B5V 71520487 IC50 > 33000 nM T42724 C1HI9J 71520488 IC50 > 33000 nM T42724 C92QDP 71520489 IC50 = 18000 nM T42724 CM6DZ1 71520490 IC50 = 2700 nM T42724 CD1XT8 71520491 IC50 > 33000 nM T42724 CU23JX 71520492 IC50 = 1000 nM T42724 CSQH86 71520575 IC50 > 33000 nM T42724 C6TO3P 71520576 IC50 = 500 nM T42724 C0WC7P 71520577 IC50 = 1800 nM T42724 CZ0QX1 71520578 IC50 = 14000 nM T42724 C8G6PW 71716112 IC50 = 7700 nM T42724 COBD81 71716733 IC50 = 14000 nM T42724 CY8AS2 71717330 IC50 = 13000 nM T42724 C2TM0Z 71719149 IC50 = 4900 nM T42724 CB0WC3 71719150 IC50 = 33000 nM T42724 CL65DR 72703815 IC50 = 49 nM T42724 C1RIO3 72704621 IC50 = 96 nM T42724 C2WO0A 72704626 IC50 = 48 nM T42724 CQ0M8X 72704809 IC50 = 52 nM T42724 C4QNK3 72704812 IC50 = 41 nM T42724 CJRX40 72705004 IC50 = 66 nM T42724 CO71SX 90644551 IC50 = 39 nM T42724 CA0L5D 90644552 IC50 = 60 nM T42724 D02CZC 9879550 IC50 = 40 nM T42724 D03FAG 138598 IC50 = 70 nM T42724 D05RLR 656734 IC50 = 20 nM T42724 D06XXG 9966986 IC50 = 9 nM T42724 D06ZNX 20684851 IC50 = 13 nM T42724 D07EYJ 9814995 IC50 = 15 nM T42724 D09LVX 9798060 IC50 = 10 nM T42724 D0A4LH 602095 IC50 = 2100 nM T42724 D0F7DQ 231627 IC50 = 330 nM T42724 D0HR0O 9884397 IC50 = 14 nM T42724 D0I5YS 5068018 IC50 = 20 nM T42724 D0K1QB 20684853 IC50 = 34 nM T42724 D0N2BP 20684855 IC50 = 30 nM T42724 D0R9CF 11302540 IC50 = 10000 nM T42724 D0T5IP 24799664 IC50 = 4300 nM T42724 D0UF2B 20684857 IC50 = 14 nM T42724 D0V7RI 9880246 IC50 = 30 nM T34471 CX4KD6 10192710 IC50 = 3100 nM T34471 CBP24H 10198140 IC50 = 61 nM T34471 C5RFA9 10214532 IC50 = 38 nM T34471 C68FIU 10214568 IC50 = 3 nM T34471 C5YRO9 10236323 IC50 = 7 nM T34471 CK05UJ 10308002 IC50 = 29000 nM T34471 C73LOJ 10308062 IC50 = 4950 nM T34471 CVK4L6 10418061 IC50 = 5400 nM T34471 C8OFL4 11241046 Ki > 10000 nM T34471 CT7IR8 12110710 IC50 = 5700 nM T34471 C6SV1C 44387258 IC50 = 2700 nM T34471 C6CT7P 44440388 IC50 = 1000 nM T34471 C28NTH 44440390 IC50 = 420 nM T34471 CM24UO 76871913 IC50 > 1000000 nM T34471 CBX7L2 90655303 IC50 > 1000000 nM T34471 CHZ2M5 90655305 IC50 > 1000000 nM T34471 CPH9G2 90655306 IC50 > 1000000 nM T34471 C9Z3YM 90655307 IC50 > 1000000 nM T34471 CI31SH 90655308 IC50 > 1000000 nM T34471 CIC01B 90655309 IC50 > 1000000 nM T34471 CN49KI 90655310 IC50 > 1000000 nM T34471 C5MBY1 90655311 IC50 > 1000000 nM T34471 CB3W0T 145961938 IC50 > 380000 nM T34471 D00DXB 10214441 IC50 = 1750 nM T34471 D06TJC 10192614 IC50 = 60 nM T34471 D0JD9E 194328 Ki = 2 nM T34471 D0R2PW 10214451 IC50 = 357 nM T73756 D03ZBT 11626560 IC50 > 10000 nM T73756 D0E6XR 3062316 IC50 = 4.4 nM T73756 D0OB0F 5328940 IC50 = 8.5 nM T73756 D0E3TC 44259 IC50 = 116 nM T73756 D0W7JZ 9911830 IC50 = 17.5 nM T73756 D0F8DL 176155 IC50 = 7800 nM T73756 D0Q7HO 4705 IC50 = 10200 nM T73756 D0T3ME 156422 IC50 = 160 nM T73756 CH21PG 2428 IC50 = 22000 nM T73756 CBPM40 4878 IC50 = 52000 nM T73756 CK0L4O 442514 IC50 > 10000 nM T73756 C7A4GI 739245 IC50 = 38000 nM T73756 CVK8Q7 876381 IC50 = 88000 nM T73756 CPR05O 2155046 IC50 = 106000 nM T73756 CVR60I 2157766 IC50 = 250000 nM T73756 CJ20AD 2157774 IC50 = 104000 nM T73756 CEJ24P 2157978 IC50 = 65000 nM T73756 CV4U8G 3132097 IC50 = 136000 nM T73756 C2IH0V 4639586 IC50 = 5200 nM T73756 C8VF0X 5328208 IC50 = 34000 nM T73756 CJL4X3 5353593 IC50 = 27500 nM T73756 CGHS32 9605612 IC50 = 94000 nM T73756 CF0EA3 11533187 IC50 > 50000 nM T73756 CACS26 11561968 Ki > 2000 nM T73756 CU0E8O 11690457 Ki > 2000 nM T73756 C8Z5VE 22431119 IC50 = 201000 nM T73756 C7YG1N 24759534 IC50 < 10 nM T73756 C4FZ8E 24875320 EC50 = 40 nM T73756 CBK82P 25011729 IC50 = 50 nM T73756 C5H7CB 44250138 EC50 = 40 nM T73756 C3VRO9 44557921 IC50 > 10000 nM T73756 C4MKC5 46870033 IC50 = 82 nM T73756 C0WYM1 46898022 IC50 = 10000 nM T73756 CS9G6E 50997096 IC50 > 10000 nM T73756 CEQN27 52936621 Ki > 1000 nM T73756 C09SDH 53257410 IC50 > 10000 nM T73756 CBK9Q6 53357848 IC50 > 10000 nM T73756 C8NA4L 53384644 IC50 = 7200 nM T73756 CXJ63M 59603829 IC50 = 36 nM T73756 CQEU96 59603842 IC50 = 2.9 nM T73756 C1MR8Q 60097495 IC50 > 1000 nM T73756 C9ZCT2 62705065 IC50 > 1000 nM T73756 CV63UL 67240318 IC50 > 10000 nM T73756 C5DGR9 69036886 IC50 = 2158 nM T73756 CPG3A5 86302574 IC50 > 30000 nM T73756 C1HW4B 89735655 IC50 = 3800 nM T73756 CPGV73 101884319 IC50 > 2000 nM T73756 CA1TZ3 101884321 IC50 > 2000 nM T73756 CG9KE7 101884322 IC50 > 2000 nM T73756 C84MVD 101884325 IC50 = 880 nM T73756 CQCX41 118737057 IC50 = 26 nM T73756 C8U0ZH 118737468 IC50 = 26.8 nM T73756 CB0QF4 122183083 IC50 > 2000 nM T73756 CB2VY7 122183099 IC50 = 2900 nM T73756 CZ1U4R 122183100 IC50 = 2200 nM T73756 C4X7SD 122192466 IC50 > 10000 nM T73756 C9WGB8 127035904 IC50 = 5400 nM T73756 CERS64 132937256 IC50 > 30000 nM T73756 CYL5V1 134694986 IC50 > 30000 nM T73756 C81FNB 135418649 IC50 = 230000 nM T73756 CY1Q3N 135438929 IC50 = 220000 nM T73756 D02NNT 53232451 IC50 > 10000 nM T73756 D02XWJ 2049 IC50 = 110000 nM T73756 D03XDN 4709 IC50 = 180000 nM T73756 D05FXD 44478401 IC50 = 1.2 nM T73756 D0C6KI 5329006 IC50 = 8500 nM T73756 D0KH5T 5687 IC50 = 1200 nM T73756 D0U2QT 1474853 IC50 = 86000 nM T73756 D0X8BU 71718651 IC50 = 3800 nM T76454 D0A7MY 637568 EC50 = 5110 nM T76454 C2UAY1 10455 IC50 > 100000 nM T76454 CKT98D 206035 IC50 > 100000 nM T76454 C9LYF4 286388 IC50 > 25000 nM T76454 CHCF90 665797 IC50 = 3000 nM T76454 CUHT06 899644 IC50 > 25000 nM T76454 CR5D2O 1070170 IC50 > 100000 nM T76454 COY71L 1073725 IC50 = 1800 nM T76454 CAP82W 1103353 IC50 > 25000 nM T76454 CG6UE9 1358452 IC50 = 2800 nM T76454 C60USN 1367926 IC50 > 25000 nM T76454 C9BPG3 1381629 IC50 = 890 nM T76454 CI5C4F 2133805 EC50 = 2900 nM T76454 CL8I0S 2772227 IC50 > 100000 nM T76454 C45EWL 3307826 EC50 > 100000 nM T76454 CXP4D9 6875758 EC50 = 9800 nM T76454 CCDG85 7514662 EC50 = 1120 nM T76454 C7GXT1 8814789 EC50 = 1060 nM T76454 CE2H5T 8814806 EC50 = 1770 nM T76454 CAH31D 8827213 EC50 = 1460 nM T76454 C4PX7O 9815648 IC50 > 100000 nM T76454 CHEX59 10329524 IC50 > 100000 nM T76454 CU79FN 16328219 EC50 = 1460 nM T76454 C1KP4N 40482356 IC50 = 2300 nM T76454 C8FD7E 40482358 EC50 > 100000 nM T76454 CZQ64N 44787480 IC50 > 25000 nM T76454 C8Z3UM 45040448 IC50 > 100000 nM T76454 C3EW7A 50744391 EC50 = 118000 nM T76454 C7PZ9N 56840728 EC50 = 2300 nM T76454 CYVK20 60149024 IC50 = 50118.72 nM T76454 C5HC3B 71681615 IC50 = 22 nM T76454 C3FVN4 71772353 IC50 > 100000 nM T76454 CK3SA1 71812184 EC50 = 1360 nM T76454 C6KD9Z 72189661 EC50 = 2420 nM T76454 C8IB1P 72189966 EC50 = 1630 nM T76454 C1LT8Q 72189968 EC50 = 2060 nM T76454 CS4QL7 72189970 EC50 = 2430 nM T76454 CAN4Z5 72771091 IC50 = 7400 nM T76454 CP7H8X 72771092 IC50 = 750 nM T76454 C38YIA 72771096 IC50 = 1100 nM T76454 C4O1IR 73330369 IC50 = 29 nM T76454 C82RVX 75202265 IC50 > 100000 nM T76454 CH9R1G 77461035 EC50 = 28.6 nM T76454 CBR20Z 91885637 IC50 = 63 nM T76454 CZ8YW7 96002439 EC50 = 5000 nM T76454 CXR0O8 106325804 IC50 > 100000 nM T76454 CXD39Z 118170767 EC50 = 12 nM T76454 C58FEG 118735935 IC50 = 750 nM T76454 CY3QN9 119057445 IC50 = 6200 nM T76454 C1U5AZ 122184660 IC50 = 980 nM T76454 CWY1V7 122184773 IC50 = 966 nM T76454 C1KQ4F 122184774 IC50 = 1666 nM T76454 CBS41H 122184775 IC50 = 10170 nM T76454 C60DTL 122184776 IC50 = 602 nM T76454 C2LR8K 122184777 IC50 = 18.1 nM T76454 C21HBC 122184778 IC50 = 54.3 nM T76454 CI2EZ4 122184779 IC50 = 42.3 nM T76454 CJ07IS 122184780 IC50 = 36.5 nM T76454 CF2MP3 122184781 IC50 = 14.4 nM T76454 CA2T7W 122184782 IC50 = 50.2 nM T76454 CP5NL4 122184783 IC50 = 979 nM T76454 C0OT6L 122184784 IC50 = 34.3 nM T76454 C1MG4H 122184785 IC50 = 179 nM T76454 C47JOU 122184786 IC50 = 47.4 nM T76454 CB9WT4 122184787 IC50 = 122 nM T76454 C1ISB2 122184788 IC50 = 66.1 nM T76454 CR4W6T 122184789 IC50 = 118 nM T76454 CHXM60 122184790 IC50 = 42.2 nM T76454 CL4WB3 122184791 IC50 = 1860 nM T76454 CP9N7W 122190547 EC50 = 5400 nM T76454 CKX08N 122190548 EC50 = 17100 nM T76454 CZL7X3 122190554 EC50 = 11500 nM T76454 CADN59 122190579 EC50 = 20600 nM T76454 C8FU3D 122190580 EC50 = 10000 nM T76454 C1B9FH 122190581 EC50 = 37800 nM T76454 CHS9C4 122190582 EC50 = 22600 nM T76454 C1IXV8 122190583 EC50 = 15000 nM T76454 CR48TK 122190584 EC50 = 11300 nM T76454 C1ID6T 122190585 EC50 = 15000 nM T76454 C96VNR 122190586 EC50 = 38500 nM T76454 C6UNI5 122190587 EC50 = 12700 nM T76454 CMCH49 122190589 EC50 = 8800 nM T76454 C4VK5C 122190590 EC50 = 24500 nM T76454 COC0V8 122190591 EC50 = 7100 nM T76454 C9G2JO 122194678 IC50 = 630 nM T76454 C3TG7O 122194679 IC50 > 25000 nM T76454 C4G5CV 122194680 IC50 > 25000 nM T76454 CPN19J 122194681 IC50 = 1100 nM T76454 CKT2A0 122194682 IC50 = 190 nM T76454 C4U7RN 122194683 IC50 = 660 nM T76454 CE45IP 122194684 IC50 > 25000 nM T76454 C2P8GB 122194685 IC50 > 25000 nM T76454 CA06HT 122194686 IC50 > 25000 nM T76454 CEI45M 122194687 IC50 > 25000 nM T76454 CNOL81 122194688 IC50 > 25000 nM T76454 CQ7NK0 122194689 IC50 > 25000 nM T76454 C9B5FT 122194690 IC50 > 25000 nM T76454 C5D3PT 122194808 IC50 > 25000 nM T76454 CJ28CN 122194809 IC50 = 410 nM T76454 C4KPW8 122194810 IC50 = 85 nM T76454 CLX1H2 122194811 IC50 > 25000 nM T76454 CB7DW0 122194812 IC50 > 25000 nM T76454 C5WZ9F 122194813 IC50 > 25000 nM T76454 CCVQ94 122194814 IC50 > 25000 nM T76454 CT0Q6I 122194815 IC50 = 5500 nM T76454 CGPU04 122194816 IC50 > 25000 nM T76454 C2RUM6 122194817 IC50 > 25000 nM T76454 C6H8SZ 126754132 IC50 < 10 nM T76454 CVL17P 134135178 IC50 = 320 nM T76454 C8IN5B 134139769 IC50 = 875 nM T76454 CLAP94 134141598 IC50 = 200 nM T76454 C9KCA0 134141909 IC50 = 230 nM T76454 CE8SA7 134145193 IC50 = 720 nM T76454 CT62RW 134148665 IC50 = 1300 nM T76454 CSW15J 134150874 IC50 = 634 nM T76454 C28GDW 134152173 IC50 = 3200 nM T76454 CU75YM 134155904 IC50 = 150 nM T76454 C0AG9Z 134813907 IC50 = 60 nM T76454 C85BCI 145951631 IC50 = 1100 nM T76454 CWKC32 145951903 IC50 > 25000 nM T76454 CJPS35 145952403 IC50 > 25000 nM T76454 C4XK3E 145952882 IC50 > 25000 nM T76454 C9N2PW 145952907 IC50 = 101 nM T76454 CIR3D0 145954661 IC50 = 1300 nM T76454 CR67LU 145955145 IC50 = 69700 nM T76454 CW3F9D 145956525 IC50 > 25000 nM T76454 C6UI5X 145956930 IC50 > 25000 nM T76454 CLG56Z 145957104 IC50 > 25000 nM T76454 C0T7QR 145971211 IC50 > 25000 nM T76454 CXLJ15 145973160 IC50 > 25000 nM T76454 CHO10Y 145974303 IC50 > 100000 nM T76454 C5OL0F 145975241 EC50 = 79 nM T76454 CD6L1Q 145979081 IC50 > 100000 nM T76454 CY6PF7 146680922 IC50 = 15.8 nM T76454 CJG46A 155510853 IC50 = 63095.73 nM T76454 C9VYG6 155511125 IC50 > 100000 nM T76454 CUY3M5 155511349 IC50 > 100000 nM T76454 CR01LK 155513180 IC50 = 50118.72 nM T76454 C7ON3W 155513257 IC50 = 19952.62 nM T76454 CK0R4I 155514102 IC50 > 100000 nM T76454 CJ3WP0 155514543 EC50 = 1390 nM T76454 CO9RY3 155515282 IC50 = 50118.72 nM T76454 CUT94K 155515491 EC50 = 970 nM T76454 CTJ97K 155516643 IC50 > 100000 nM T76454 CT28RK 155516991 IC50 = 39810.72 nM T76454 CC9K7R 155517070 IC50 = 50118.72 nM T76454 CYD95J 155517097 IC50 = 39810.72 nM T76454 CP68KM 155517263 IC50 = 50118.72 nM T76454 CB9MT8 155519311 IC50 = 15848.93 nM T76454 C68RTM 155519428 EC50 = 1360 nM T76454 CE6S0K 155519779 IC50 = 6309.57 nM T76454 C9TFN3 155520145 IC50 = 50118.72 nM T76454 C7PO4L 155520368 EC50 = 1910 nM T76454 CYX39S 155520897 EC50 = 1100 nM T76454 CUWL37 155521263 EC50 = 990 nM T76454 CA8IS0 155521928 IC50 = 19952.62 nM T76454 CL65ZK 155524194 IC50 > 100000 nM T76454 CS0WI3 155525300 IC50 = 2600 nM T76454 C73KQP 155525472 IC50 = 39810.72 nM T76454 C3MDZ4 155525522 IC50 > 100000 nM T76454 C4BAY9 155526259 IC50 > 100000 nM T76454 C8JU0Y 155526260 IC50 > 100000 nM T76454 C5RPQ3 155526688 IC50 > 100000 nM T76454 CJX51W 155527016 IC50 > 100000 nM T76454 C90REN 155527528 EC50 = 630 nM T76454 CEP71W 155528033 IC50 = 5011.87 nM T76454 CWI4Q5 155528195 IC50 = 50118.72 nM T76454 CCE2M5 155528362 IC50 > 100000 nM T76454 CS3QI5 155528453 EC50 = 3330 nM T76454 CFO37K 155528822 IC50 = 15848.93 nM T76454 C7L6CB 155529157 IC50 = 12589.25 nM T76454 C38UVP 155529704 IC50 = 12589.25 nM T76454 CKGA51 155530132 IC50 > 100000 nM T76454 C1ZTY3 155530152 IC50 = 63095.73 nM T76454 CEJQ10 155530334 IC50 = 3981.07 nM T76454 CQ4OC5 155531518 IC50 > 100000 nM T76454 CD5B4Z 155531917 IC50 > 100000 nM T76454 CCZ13G 155532065 IC50 = 50118.72 nM T76454 CU1A8Y 155532391 IC50 > 100000 nM T76454 C23ISL 155533277 EC50 = 1230 nM T76454 C7Q8UV 155533600 EC50 = 1540 nM T76454 CPH14B 155533997 IC50 > 50000 nM T76454 C2ZX3Y 155534140 EC50 = 2580 nM T76454 CWQ8P2 155534356 EC50 > 5000 nM T76454 C3K4EL 155535225 IC50 = 5011.87 nM T76454 C0Y9OK 155536020 IC50 = 39810.72 nM T76454 CF36VE 155536250 IC50 = 31622.78 nM T76454 COZC62 155536474 IC50 = 15848.93 nM T76454 CC64FE 155536577 IC50 = 50118.72 nM T76454 CO6ER7 155537046 IC50 = 25118.86 nM T76454 CW7AK4 155537439 IC50 = 15848.93 nM T76454 CK62ID 155537869 IC50 > 100000 nM T76454 C3WE9N 155538368 IC50 = 31622.78 nM T76454 C2RS7E 155539746 IC50 = 609 nM T76454 C75KYA 155540072 IC50 = 19952.62 nM T76454 C6PTE5 155540447 IC50 = 10000 nM T76454 CF0RT5 155540699 IC50 > 100000 nM T76454 CPFC16 155540797 IC50 = 63095.73 nM T76454 C67XKR 155541172 IC50 = 50118.72 nM T76454 C1L0WK 155541675 IC50 > 100000 nM T76454 C43NZV 155542200 IC50 = 10000 nM T76454 CQ8PW0 155542328 IC50 > 100000 nM T76454 CF2P7M 155542638 IC50 > 100000 nM T76454 C4MOF9 155543478 IC50 > 100000 nM T76454 CX8YP9 155543849 EC50 > 5000 nM T76454 C4G6RN 155544017 EC50 > 1000 nM T76454 C2M7EI 155544159 IC50 = 25118.86 nM T76454 C6JOP4 155545387 IC50 = 5011.87 nM T76454 C7UD2J 155546696 IC50 = 50118.72 nM T76454 CZ0I1S 155547074 IC50 > 100000 nM T76454 CQBT74 155547935 IC50 = 19952.62 nM T76454 CO7G5S 155548430 IC50 > 100000 nM T76454 C5XD8R 155548655 IC50 > 100000 nM T76454 C1V5OY 155548738 EC50 = 5520 nM T76454 CEPW05 155549226 IC50 = 100000 nM T76454 CT20GV 155549977 IC50 = 10000 nM T76454 CV4PU6 155550024 IC50 > 50000 nM T76454 CQ1TK8 155550838 EC50 = 1720 nM T76454 C5L8JE 155552136 IC50 > 100000 nM T76454 C9P1KN 155552525 IC50 > 50000 nM T76454 CDK9G7 155553288 IC50 = 2511.89 nM T76454 CH4G2N 155553767 IC50 > 100000 nM T76454 C8YIK6 155553920 IC50 = 25118.86 nM T76454 CNS6W1 155554404 EC50 = 1800 nM T76454 CBQ1U7 155554694 EC50 = 6970 nM T76454 CX83BF 155555686 IC50 = 39810.72 nM T76454 C6WPD1 155555697 IC50 = 50118.72 nM T76454 C0BPZ3 155555710 IC50 = 7943.28 nM T76454 C93OHG 155556364 IC50 = 31622.78 nM T76454 C8BQE6 155556461 IC50 = 15848.93 nM T76454 CQS7P0 155557407 IC50 = 39810.72 nM T76454 CB8Q5Y 155557794 IC50 = 12589.25 nM T76454 CL9F3S 155557868 IC50 = 25118.86 nM T76454 CRL16T 155558461 IC50 = 39810.72 nM T76454 C9XCN2 155558691 IC50 = 31622.78 nM T76454 C1C0ZO 155560119 EC50 = 2840 nM T76454 C24WDN 155560460 IC50 > 100000 nM T76454 CP2H0X 155560853 IC50 > 100000 nM T76454 CB63KG 155561425 IC50 > 100000 nM T76454 CEY87B 155562396 IC50 > 50000 nM T76454 CIJ0H9 155562696 IC50 > 100000 nM T76454 CB6NP3 155563580 IC50 = 31622.78 nM T76454 C13OYN 155563808 IC50 = 31622.78 nM T76454 CP61RM 155564286 IC50 = 31622.78 nM T76454 CA1K9B 155564526 IC50 = 7943.28 nM T76454 C4AL7M 155564597 IC50 > 100000 nM T76454 C85CMZ 155564705 IC50 = 25118.86 nM T76454 C1GUE5 155564896 EC50 = 2300 nM T76454 C6O4NA 155566445 IC50 = 25118.86 nM T76454 CF32ZO 155566614 IC50 > 100000 nM T76454 CC1H8N 155569160 IC50 > 50000 nM T76454 C5P6OE 155569644 IC50 > 100000 nM T76454 D0X4IO 5350 EC50 = 870 nM T92458 D00DYK 10672195 IC50 = 27 nM T92458 D08UGX 60652 IC50 = 2.3 nM T92458 C9LCD8 3823 Ki = 33 nM T92458 CXQ40P 5862285 IC50 = 480100 nM T92458 CKP8J2 9952928 IC50 = 15 nM T92458 C2NC9T 9982688 IC50 = 549 nM T92458 CO6SL8 10006229 IC50 = 28 nM T92458 C0AIR8 10254192 IC50 = 13 nM T92458 CSF9D6 10436341 IC50 = 20.5 nM T92458 CSKJ13 10476195 IC50 = 15.1 nM T92458 C4GO0T 11231328 IC50 = 900 nM T92458 CW51VQ 11523005 IC50 = 122000 nM T92458 CM23NT 11627214 IC50 = 28 nM T92458 C8OCK9 44445025 IC50 = 7.4 nM T92458 CIGH93 46913220 IC50 = 4000 nM T92458 CX06UZ 46913221 IC50 = 2800 nM T92458 COJR54 46913222 Ki = 28 nM T92458 C2OVH8 46945071 IC50 = 11220 nM T92458 CZU4R8 46945072 IC50 = 10760 nM T92458 CQY49U 46945073 IC50 = 2080 nM T92458 C40UXW 46945265 IC50 = 16300 nM T92458 CUND25 46945267 IC50 = 5080 nM T92458 C21XOI 46945268 IC50 = 127600 nM T92458 CYJ6B3 46945269 IC50 = 342800 nM T92458 CVM1X7 46945270 IC50 = 25570 nM T92458 C8SAD4 46945450 IC50 = 1920 nM T92458 C3Y1MH 49798926 IC50 = 36900 nM T92458 C3H0OP 49798927 IC50 = 6400 nM T92458 CAG5E4 49798928 IC50 = 10600 nM T92458 CSL4W6 49798929 IC50 = 23000 nM T92458 CDT94F 49798930 IC50 = 72000 nM T92458 CP0Z4I 52947291 IC50 = 111100 nM T92458 CN2U4D 71470821 Ki = 42 nM T92458 CKB74E 101563630 Ki = 21 nM T92458 C65OBE 102263901 Ki = 39 nM T92458 C08MUX 118712539 Ki = 19 nM T92458 CIJ8X3 118712540 Ki = 24 nM T92458 CB4RF3 118712541 Ki = 7.8 nM T92458 C7R0HI 118712542 Ki = 9.7 nM T92458 C2GY4L 118712543 Ki = 36 nM T92458 C4BF0D 118712544 Ki = 91 nM T92458 C2G0IS 118712545 Ki = 150 nM T92458 C7GW1F 118712546 Ki = 11 nM T92458 CVA28S 118712547 Ki = 400 nM T92458 CT3K0P 118712548 Ki = 380 nM T92458 C15VDJ 118712549 Ki = 210 nM T92458 CQ17VZ 118712550 Ki = 13 nM T92458 CM02GX 118712551 Ki = 42 nM T92458 C9PHX0 118717751 Ki = 26 nM T92458 C2U3PM 118717752 Ki = 31 nM T92458 C0N3SH 118717753 Ki = 14 nM T92458 C1LH3Q 118717754 Ki = 14 nM T92458 COEC25 118717755 Ki = 37 nM T92458 C28TZN 118717756 Ki = 37 nM T92458 C9L3FI 118717757 Ki = 340 nM T92458 C7LO3N 118717758 Ki = 730 nM T92458 CFV32P 118717759 Ki = 230 nM T92458 C2UKD8 118717760 Ki = 740 nM T92458 CT41OR 118717761 Ki = 540 nM T92458 CM7YZ6 118717762 Ki = 640 nM T92458 C29QXN 118717763 Ki = 1190 nM T92458 C4JK3Y 132576469 IC50 = 180 nM T92458 C2A7XR 132576470 IC50 = 350 nM T92458 CJ3G1E 132576471 IC50 = 110 nM T92458 CRX9U7 132576473 IC50 = 340 nM T92458 C8SMW6 132576474 IC50 = 190 nM T92458 CA26QP 132576475 IC50 = 150 nM T92458 CJ0AW5 137642065 IC50 = 160 nM T92458 CK85HZ 137642698 IC50 = 210 nM T92458 CUV6R4 137646382 IC50 = 120 nM T92458 C5L4DT 137647630 IC50 = 4480 nM T92458 C8BVR4 137650145 IC50 = 2600 nM T92458 CSR6M7 137651189 IC50 = 310 nM T92458 CSJ4F6 137658543 IC50 = 2500 nM T92458 C91SEX 137659282 IC50 > 10000 nM T92458 D04UAZ 9982767 IC50 = 6.5 nM T75136 CYG60X 512874 Ki = 81.4 nM T75136 CBL1C6 10883540 EC50 = 430 nM T75136 C8C9HM 11132282 EC50 = 22 nM T75136 CB96ZX 24742075 Ki = 64.3 nM T75136 CYL7A6 24825421 EC50 = 90 nM T75136 CI38DG 24825422 EC50 = 12 nM T75136 C5T6WY 24825423 EC50 = 160 nM T75136 CB8EU6 24825424 EC50 = 100 nM T75136 CN5Q0O 24825425 EC50 = 60 nM T75136 CWQU39 24825426 EC50 = 1400 nM T75136 C5EIS2 24825427 EC50 > 10000 nM T75136 CH3YB9 24825428 EC50 = 70 nM T75136 C9NPK4 24825429 EC50 = 320 nM T75136 C7OI1S 24825430 EC50 = 2100 nM T75136 CXRQ34 24825431 EC50 = 31.62 nM T75136 C4WTY2 24825432 EC50 = 230 nM T75136 C9ZDA7 24825433 EC50 > 10000 nM T75136 CLW5C7 24825434 EC50 = 150 nM T75136 CFV48O 24825435 EC50 = 330 nM T75136 C2FKX4 24825436 EC50 = 1000 nM T75136 CV25CA 24825437 EC50 = 30 nM T75136 COM6B8 24825438 EC50 > 10000 nM T75136 CYM47L 24825439 EC50 > 10000 nM T75136 CK4AB0 24825440 EC50 > 10000 nM T75136 CN84ZX 24825441 EC50 = 1200 nM T75136 C4RS1G 52936713 EC50 = 251.19 nM T75136 CA15HU 52936816 EC50 = 398.11 nM T75136 C6BH1V 52936819 EC50 = 1000 nM T75136 CRY03J 52936822 EC50 = 2511.89 nM T75136 CWRU85 52936928 EC50 = 2511.89 nM T75136 CF7M2A 52936929 EC50 = 3162.28 nM T75136 C2GV4R 52936930 EC50 = 5011.87 nM T75136 CAT2L4 52936931 EC50 = 2511.89 nM T75136 COLN94 52936934 EC50 = 794.33 nM T75136 CR6HC7 52937033 EC50 = 100 nM T75136 C2TI8L 52937034 EC50 = 251.19 nM T75136 CCWO80 52937035 EC50 = 316.23 nM T75136 CJ6K7I 52937037 EC50 = 1995.26 nM T75136 CI4Q9R 52937137 EC50 = 1000 nM T75136 CY10CO 52937140 EC50 = 3162.28 nM T75136 C6W5GH 52937141 EC50 = 2511.89 nM T75136 CENW79 52937246 EC50 = 251.19 nM T75136 C7I0MG 52937350 EC50 = 1258.93 nM T75136 CJ3E9B 52937351 EC50 = 794.33 nM T75136 CKC03F 52937353 EC50 = 199.53 nM T75136 CO6AG4 52937354 EC50 = 1584.89 nM T75136 CM7UT9 52937355 EC50 = 158.49 nM T75136 C45YZW 52937356 EC50 = 1258.93 nM T75136 CG98BX 52937447 EC50 = 316.23 nM T75136 CX32GP 52937449 EC50 = 398.11 nM T75136 CING80 52937450 EC50 = 251.19 nM T75136 C68SHU 52937451 EC50 = 1584.89 nM T75136 CHOZ17 52937452 EC50 = 501.19 nM T75136 CL96WV 54580360 EC50 = 251.19 nM T75136 CC67DZ 126673332 Ki = 7000 nM T75136 C16CVG 138857911 EC50 = 600 nM T75136 C0NF4Q 138857912 EC50 = 15 nM T75136 CRFJ45 138857913 EC50 = 13000 nM T75136 CZ93GB 139030532 Ki = 2.1 nM T75136 CE3T1J 145984173 EC50 = 13000 nM T75136 C36QJH 145988910 EC50 = 5000 nM T75136 C97VJP 145990098 EC50 = 400 nM T75136 C0AIB6 155518824 EC50 = 40 nM T75136 C94IEB 155522101 Ki = 2400 nM T75136 CN7HV4 155522503 EC50 = 900 nM T75136 CTR04M 155524650 EC50 = 800 nM T75136 CF3P4T 155527718 EC50 = 1000 nM T75136 C7LHO4 155535510 EC50 = 2000 nM T75136 C91LUA 155539274 EC50 = 9000 nM T75136 CR8AY9 155545328 EC50 = 5000 nM T75136 CG4QF6 155551225 EC50 = 500 nM T75136 C96DYA 155554234 EC50 = 100 nM T75136 CTX5J9 155557666 EC50 = 800 nM T75136 CD8TS3 155558831 EC50 = 3000 nM T75136 CJF3I2 155564002 EC50 = 4000 nM T08922 D03KHO 52934180 IC50 = 33 nM T08922 D04SOU 24964679 IC50 = 3 nM T08922 CR6J9X 1346344 IC50 = 3600 nM T08922 CTM96E 2258378 IC50 = 359 nM T08922 C8Y6BN 8072533 IC50 = 6600 nM T08922 C0XU7G 11516410 IC50 = 11 nM T08922 CLE5T1 11537493 IC50 = 4 nM T08922 COC70H 11552248 IC50 = 69 nM T08922 CB1R6F 11559272 IC50 = 15 nM T08922 CNR1F7 11587962 IC50 = 1860 nM T08922 CHCE80 11588060 IC50 = 2420 nM T08922 CO52NA 11595374 IC50 = 19 nM T08922 C7FHT4 11609746 IC50 = 6 nM T08922 C9UK3N 11631866 IC50 = 96 nM T08922 CWF5L3 11638609 IC50 = 600 nM T08922 CKC2G7 11674600 IC50 > 30000 nM T08922 C3SMK1 11674889 IC50 = 30 nM T08922 CPY92G 11681998 IC50 = 38 nM T08922 C1DGX2 11682005 IC50 = 55 nM T08922 CH4VD1 11682200 IC50 = 840 nM T08922 CIK8R6 11696186 IC50 = 1510 nM T08922 CB9H6C 11702917 IC50 = 150 nM T08922 CSD2O8 11716889 IC50 > 30000 nM T08922 CYM4J0 11717830 IC50 = 26 nM T08922 CC8W6L 16049279 IC50 = 13 nM T08922 CI06KZ 16049349 IC50 = 33 nM T08922 CU3V4D 16049419 IC50 = 23 nM T08922 C9U1QI 16049420 IC50 = 40 nM T08922 CEBC71 16049422 IC50 = 18 nM T08922 CPV58U 16049424 IC50 = 49 nM T08922 CI4B3V 16066829 IC50 = 37 nM T08922 CCE42Y 16110742 IC50 > 30000 nM T08922 CO9CX8 16110743 IC50 = 14 nM T08922 CB3H7E 16110744 IC50 = 26 nM T08922 C8OID1 16110748 IC50 = 8 nM T08922 CN2KC3 16110750 IC50 = 3 nM T08922 C1N9KY 16110753 IC50 = 28 nM T08922 CRE71K 16110754 IC50 = 7 nM T08922 C16FVA 16110755 IC50 = 47 nM T08922 C7E3UV 16110756 IC50 = 9 nM T08922 CC98WT 16110757 IC50 = 630 nM T08922 C9X1UF 16730599 IC50 = 13 nM T08922 C14KRF 16747776 IC50 = 12000 nM T08922 CEHK12 24957986 IC50 = 400 nM T08922 CROK95 24958582 IC50 = 14 nM T08922 CTC4N7 24958944 IC50 = 16 nM T08922 C2I7PV 24958946 IC50 = 27 nM T08922 C7SF3X 25124945 IC50 = 110 nM T08922 C0HLZ8 44125793 IC50 = 2900 nM T08922 C7VOU1 44126023 IC50 = 52 nM T08922 CF1LV2 44126025 IC50 = 4500 nM T08922 CXF12E 44126528 IC50 = 210 nM T08922 CR80JA 44199807 IC50 = 20 nM T08922 C5X4ZH 44199810 IC50 = 8.1 nM T08922 CFA27C 44199917 IC50 = 33 nM T08922 CC03TW 44199919 IC50 = 36 nM T08922 C3TZ4U 44199920 IC50 = 23 nM T08922 CE0K5B 44200032 IC50 = 6.1 nM T08922 CCF6J7 44200033 IC50 = 4.9 nM T08922 C6M1WI 44420147 IC50 = 57 nM T08922 CL4P8A 44420148 IC50 = 290 nM T08922 C5CFJ3 44420152 IC50 = 1620 nM T08922 C0YOV9 44420159 IC50 > 30000 nM T08922 CT7LW3 44420165 IC50 = 26500 nM T08922 CD5C0L 44420173 IC50 > 30000 nM T08922 CS5Y8F 44420174 IC50 = 370 nM T08922 C3W4PD 44420185 IC50 = 67 nM T08922 CQ84PI 44420191 IC50 = 4050 nM T08922 CG6U1C 44420195 IC50 = 81 nM T08922 CCD3F6 44420197 IC50 = 340 nM T08922 CBZ4V5 44420200 IC50 = 76 nM T08922 C3AB7C 44420201 IC50 = 19480 nM T08922 CADL51 44420204 IC50 = 130 nM T08922 C0RVQ4 44420205 IC50 = 1320 nM T08922 CWSC52 44420206 IC50 = 350 nM T08922 C3X4RK 44420208 IC50 = 1310 nM T08922 C1QVU7 44420209 IC50 = 6160 nM T08922 CT7BN1 44420210 IC50 = 1960 nM T08922 C0KLB6 44420211 IC50 = 380 nM T08922 C17QEG 44420213 IC50 = 1700 nM T08922 CY3TS2 44420214 IC50 = 470 nM T08922 C28LXO 44420216 IC50 = 850 nM T08922 CN46XM 44420217 IC50 = 10 nM T08922 C3D8BO 44420220 IC50 = 13 nM T08922 COD9K2 44420221 IC50 = 16 nM T08922 CS7X2F 44420223 IC50 = 5 nM T08922 CZ9J8E 44420224 IC50 = 27 nM T08922 CJ9F2V 44420229 IC50 > 30000 nM T08922 CFO87J 44420230 IC50 > 30000 nM T08922 C5U7BP 44420289 IC50 = 14 nM T08922 CO9G0R 44420292 IC50 = 26 nM T08922 C2M3SL 44420295 IC50 = 210 nM T08922 C9MHV7 44431784 IC50 = 18 nM T08922 CZR60X 44431785 IC50 > 30000 nM T08922 C72IJO 44431786 IC50 = 260 nM T08922 CIUH67 44431787 IC50 = 1000 nM T08922 CY8E3N 44431789 IC50 = 42 nM T08922 CTZ6I2 44431790 IC50 = 15800 nM T08922 C0QY2O 44431791 IC50 > 30000 nM T08922 CKQ02Z 44431792 IC50 = 550 nM T08922 C9AEM5 44431793 IC50 = 9 nM T08922 C2DUA3 44431794 IC50 = 70 nM T08922 C1I5WV 44431795 IC50 = 140 nM T08922 C5O1KF 44431796 IC50 = 11 nM T08922 CDZ2O0 44431797 IC50 = 35 nM T08922 CE95OL 44431798 IC50 = 34 nM T08922 C0PD9Q 44431799 IC50 = 29 nM T08922 CQ4EV3 44431800 IC50 = 13 nM T08922 C8TF7P 44431801 IC50 = 10 nM T08922 CGE71U 44431804 IC50 = 69 nM T08922 CGCR90 44431805 IC50 = 12 nM T08922 CU75RY 44442774 IC50 = 690 nM T08922 C1RET0 44442775 IC50 > 30000 nM T08922 C52EZC 44442776 IC50 = 42 nM T08922 C51IMO 44442778 IC50 = 3980 nM T08922 CV32WG 44442779 IC50 = 83 nM T08922 C8LQO6 44442781 IC50 = 57 nM T08922 CQR90Z 44442782 IC50 = 38 nM T08922 CJUZ92 44442784 IC50 = 440 nM T08922 C04YWO 44442787 IC50 = 37 nM T08922 C1N8YK 44442789 IC50 = 71 nM T08922 CXQ47M 44442790 IC50 = 330 nM T08922 CZ5UX0 44442792 IC50 = 670 nM T08922 C1N6DH 44442794 IC50 = 680 nM T08922 CV0Z5D 44442795 IC50 = 20490 nM T08922 CIA7E2 44442796 IC50 = 920 nM T08922 C5O1LP 44442797 IC50 = 850 nM T08922 CPWQ62 44442798 IC50 > 30000 nM T08922 CNS3K8 44442799 IC50 = 570 nM T08922 CD20FT 44442800 IC50 = 220 nM T08922 CR4BE6 44442801 IC50 > 30000 nM T08922 CF3SQ0 44442802 IC50 = 500 nM T08922 C9D4RJ 44442804 IC50 = 530 nM T08922 CH2K3X 44442808 IC50 = 910 nM T08922 C6O0ZQ 44476624 IC50 = 9.8 nM T08922 CNI0E4 44519497 IC50 = 13 nM T08922 C5AI0L 44519498 IC50 = 14 nM T08922 CPDG26 44519663 IC50 = 29 nM T08922 C20CIE 44554862 IC50 = 30 nM T08922 C6N3LY 44608464 IC50 = 140 nM T08922 CX69HR 44608465 IC50 = 190 nM T08922 CD92FW 44608467 IC50 = 400 nM T08922 CF74VQ 44608621 IC50 = 1280 nM T08922 CMVG38 44608622 IC50 = 210 nM T08922 CP97QX 44608623 IC50 = 200 nM T08922 C0CQO9 44608787 IC50 = 70 nM T08922 C4D9PW 44610762 IC50 = 119 nM T08922 CT42CD 44610763 IC50 = 14 nM T08922 CVTP57 44610765 IC50 = 7 nM T08922 CGZ8D1 44610766 IC50 = 945 nM T08922 C2I5GM 44610767 IC50 = 30000 nM T08922 CC9PH2 44610768 IC50 = 373 nM T08922 C7HJ9O 44610769 IC50 = 102 nM T08922 CNE4T3 45100495 IC50 = 641 nM T08922 CD8B0J 45375926 IC50 = 23 nM T08922 C6FO0S 45487686 IC50 = 718 nM T08922 C5O7PA 45487687 IC50 = 1840 nM T08922 CH82OC 45487688 IC50 = 35 nM T08922 CS76MT 45487690 IC50 = 12 nM T08922 C74GYW 45487691 IC50 = 550 nM T08922 CUK5X6 45487700 IC50 = 141 nM T08922 CR2GA9 45487701 IC50 = 1510 nM T08922 C5NY7X 45487709 IC50 = 114 nM T08922 CB57IT 45487710 IC50 = 609 nM T08922 CX1H3A 45487711 IC50 = 3100 nM T08922 CYE81D 45487712 IC50 = 881 nM T08922 CK74PQ 45487713 IC50 = 2540 nM T08922 CY40OH 45487721 IC50 = 35 nM T08922 C6VRU2 45487722 IC50 = 227 nM T08922 CGXZ54 45487723 IC50 = 8 nM T08922 CNPR63 45487727 IC50 = 303 nM T08922 C1KI8Y 45487728 IC50 = 88 nM T08922 C4OK5A 45487729 IC50 = 777 nM T08922 C0OK3C 45487733 IC50 = 274 nM T08922 C3EQB4 45487734 IC50 = 18 nM T08922 C9H5KT 45487742 IC50 = 33 nM T08922 C9VNI2 45487743 IC50 = 16 nM T08922 CX6S5Z 45487744 IC50 = 202 nM T08922 CN5AD4 45487745 IC50 = 93 nM T08922 CZ34CP 45487746 IC50 = 32 nM T08922 CFE7D6 45487751 IC50 > 30000 nM T08922 CIH84V 45487752 IC50 > 30000 nM T08922 CT9OI3 45487756 IC50 = 30000 nM T08922 C35CAQ 45487757 IC50 = 117 nM T08922 C84CBM 45487758 IC50 = 494 nM T08922 CT6NS7 45487763 IC50 = 113 nM T08922 C9OHV3 45487764 IC50 = 156 nM T08922 CC6IF0 45487775 IC50 = 268 nM T08922 C8EGW1 45487776 IC50 = 214 nM T08922 C30ZTE 46830213 IC50 = 4.5 nM T08922 C57OXQ 46830214 IC50 = 20 nM T08922 C5Y4AQ 46884569 IC50 = 48 nM T08922 C2CKL7 46884570 IC50 = 6.5 nM T08922 CS2G4I 46884619 IC50 = 164 nM T08922 CVB9W3 46884621 IC50 = 151 nM T08922 CXC1J6 46884622 IC50 = 11 nM T08922 CBPW05 46884651 IC50 = 16 nM T08922 CIB15R 46884652 IC50 = 111 nM T08922 C75LXJ 46884653 IC50 = 126 nM T08922 C06LUI 46884654 IC50 > 1000 nM T08922 C9ZT2U 46884680 IC50 = 505 nM T08922 CH42ZS 46884681 IC50 = 11 nM T08922 C2YT9I 46884682 IC50 = 16 nM T08922 C6E4JQ 46884683 IC50 = 16 nM T08922 CN45YI 46884711 IC50 = 12 nM T08922 C5A0RB 46884712 IC50 = 19 nM T08922 CA15IS 46884713 IC50 = 51 nM T08922 CVU9W1 46884797 IC50 = 4.5 nM T08922 CZ1AY8 46884798 IC50 = 6.1 nM T08922 C7SA3X 46884799 IC50 = 7.6 nM T08922 CKG4R3 46884800 IC50 = 30 nM T08922 CQ2X7O 46884844 IC50 = 39 nM T08922 C92KGL 46884845 IC50 = 6.4 nM T08922 CK9FU1 46884847 IC50 = 0.3 nM T08922 C09SVP 46884881 IC50 = 0.31 nM T08922 CU38VO 46884883 IC50 = 363 nM T08922 C4IX1Z 46884885 IC50 = 640 nM T08922 CV0GE3 46884924 IC50 = 48 nM T08922 CLEK60 46884925 IC50 = 98 nM T08922 CC79WD 46885253 IC50 = 2130 nM T08922 C6AW3N 46885303 IC50 > 1000 nM T08922 CO0M3V 46885304 IC50 > 1000 nM T08922 C2V5YE 49843456 IC50 = 330 nM T08922 CP8W1J 49855399 IC50 = 670 nM T08922 CH7E9C 49855400 IC50 = 250 nM T08922 C25ATW 49855401 IC50 = 190 nM T08922 C1CZ5E 49855402 IC50 = 150 nM T08922 CB4TR0 49855404 IC50 = 60 nM T08922 CI9PJ4 49855596 IC50 = 100 nM T08922 CH6K1T 49855597 IC50 > 30000 nM T08922 C96FUO 49855598 IC50 = 200 nM T08922 C23JIY 49855599 IC50 = 7800 nM T08922 CZ3GE6 49855600 IC50 = 80 nM T08922 CMZT98 49858286 IC50 = 80 nM T08922 C7LQR8 49858287 IC50 = 700 nM T08922 C4OI0V 49858288 IC50 = 6700 nM T08922 CKDE49 52933949 IC50 = 17 nM T08922 CL2Q9F 52934178 IC50 = 30 nM T08922 C8J5MA 53316558 IC50 = 2650 nM T08922 C7L3WJ 53317443 IC50 = 95 nM T08922 C4O5QF 53319127 IC50 = 1200 nM T08922 CSK32V 53319197 IC50 = 630 nM T08922 CCI73H 53319198 IC50 = 700 nM T08922 CY7WZ2 53320341 IC50 = 270 nM T08922 C6S8NU 53320460 IC50 = 15 nM T08922 CTJ7S8 53323129 IC50 = 2100 nM T08922 C4V3HW 53325421 IC50 = 60 nM T08922 C7PI5Z 53384658 IC50 = 5.4 nM T08922 CEC38U 54104450 IC50 = 2500 nM T08922 CQ7M4A 56659186 IC50 = 690 nM T08922 C17OQE 56662690 IC50 = 1300 nM T08922 C0EF3R 56662691 IC50 = 730 nM T08922 CXFL76 56662692 IC50 = 110 nM T08922 CPB8O2 56662693 IC50 = 89 nM T08922 CA2ZV4 56666145 IC50 = 5800 nM T08922 CW6IY5 56666146 IC50 = 570 nM T08922 CSGM94 56666156 IC50 = 750 nM T08922 CF7Z8H 56669553 IC50 = 240 nM T08922 CKO8M6 56669554 IC50 = 99 nM T08922 CZ7XK8 56671907 IC50 = 1700 nM T08922 CH2D6N 56673072 IC50 = 690 nM T08922 CG9RP3 56673073 IC50 = 1400 nM T08922 C0ZB1D 56673074 IC50 = 680 nM T08922 CGAF01 56673075 IC50 = 130 nM T08922 C6U5FO 56676377 IC50 = 780 nM T08922 CK2GQ7 56679719 IC50 = 230 nM T08922 CP18ZJ 56679720 IC50 = 630 nM T08922 CP24HC 56683036 IC50 = 3800 nM T08922 C25PQT 56683037 IC50 = 210 nM T08922 C78DEZ 56949650 IC50 = 37 nM T08922 CAF78E 56949651 IC50 = 27 nM T08922 C1HUL5 56949652 IC50 = 18 nM T08922 C8ZJ1O 56949653 IC50 = 92 nM T08922 C6NI3A 56949654 IC50 = 80 nM T08922 CZ4IJ1 56949778 IC50 = 56 nM T08922 C2GNQ9 56949779 IC50 = 20 nM T08922 CR1B8F 56949780 IC50 = 7.4 nM T08922 CU4X6A 56949781 IC50 = 6.6 nM T08922 C4K2MW 56949782 IC50 = 21 nM T08922 CB6NQ5 56951516 IC50 = 650 nM T08922 CQF0G9 56951517 IC50 = 470 nM T08922 C8O2CA 56951518 IC50 = 63 nM T08922 CPV34M 56951519 IC50 = 37 nM T08922 C9JDZ7 56951520 IC50 = 45 nM T08922 C29RFV 56951521 IC50 = 23 nM T08922 C1WDQ5 56951631 IC50 = 14 nM T08922 C57JQW 56951632 IC50 = 9.4 nM T08922 C4VFX1 56951633 IC50 = 63 nM T08922 COP3S4 56951634 IC50 = 6.9 nM T08922 C37GFA 56951635 IC50 = 42 nM T08922 CS94XG 56967694 IC50 = 68 nM T08922 CQCZ78 56967888 IC50 = 76 nM T08922 CN5A4B 56967890 IC50 = 29 nM T08922 CD8W9Y 56967949 IC50 = 6.8 nM T08922 CHEB78 56967950 IC50 = 3 nM T08922 CD9K3Y 56968001 IC50 = 4 nM T08922 CD82FP 56968002 IC50 = 4.2 nM T08922 C9PLF3 56968003 IC50 = 6 nM T08922 C4MB3G 56968004 IC50 = 6 nM T08922 CVR2T4 57390226 IC50 = 140 nM T08922 CT13IH 57390227 IC50 = 1000 nM T08922 CA5IH6 57392016 IC50 = 220 nM T08922 C0K2CZ 57392017 IC50 = 750 nM T08922 C5MIY2 57392018 IC50 = 15 nM T08922 C47WPG 57393731 IC50 = 8000 nM T08922 C26BSF 57393732 IC50 = 880 nM T08922 CVU43O 57393733 IC50 = 15 nM T08922 CK67TS 57393734 IC50 = 45 nM T08922 C1FQX7 57393735 IC50 = 1600 nM T08922 CHJ0D1 57393906 IC50 = 11 nM T08922 C7SC5X 57398986 IC50 = 100 nM T08922 CUSR05 57400701 IC50 = 280 nM T08922 C8ILO6 57400702 IC50 = 43 nM T08922 CRD76K 57402473 IC50 = 110 nM T08922 CC3K2A 57402474 IC50 = 360 nM T08922 C4V8TE 57402475 IC50 = 1200 nM T08922 CZD32M 57496611 IC50 = 30 nM T08922 CV8M2B 59279752 IC50 = 15 nM T08922 C52WKX 59279790 IC50 = 17 nM T08922 CZYR95 59279807 IC50 = 15 nM T08922 C3CY0B 59373318 IC50 = 22 nM T08922 C2MQI0 59373441 IC50 = 79 nM T08922 CQJ5P9 59373484 IC50 = 17 nM T08922 C4GX7L 59373545 IC50 = 75 nM T08922 CHZ75M 59373599 IC50 = 51 nM T08922 C3SIC5 59373616 IC50 = 43 nM T08922 C7UY6F 59373726 IC50 = 32 nM T08922 C9Q3AG 59373739 IC50 = 64 nM T08922 CQ26EF 60168080 IC50 = 8.5 nM T08922 CD3C7S 67204380 IC50 = 23 nM T08922 C1UG5C 67491412 IC50 = 55 nM T08922 CQ3NU0 67491582 IC50 = 29 nM T08922 C3L7BC 67491705 IC50 = 2.3 nM T08922 C14HAP 70674463 IC50 = 10 nM T08922 CIH1L4 70674464 IC50 = 2.1 nM T08922 C43FIY 70675044 IC50 = 2.9 nM T08922 C3X0QJ 70684264 IC50 = 5.1 nM T08922 CX20NS 70687952 IC50 = 4.4 nM T08922 C0EXA5 70688510 IC50 = 8.7 nM T08922 CIQR26 70689978 IC50 = 9 nM T08922 CR1G7Z 70690580 IC50 = 5.9 nM T08922 C14RZE 70692134 IC50 = 37 nM T08922 C5NAO2 70692713 IC50 = 7.5 nM T08922 C6RBG1 71462326 IC50 = 2800 nM T08922 C0VLE3 71516457 IC50 = 13 nM T08922 C2LVY0 71516458 IC50 = 31 nM T08922 C0GVH3 71718672 IC50 = 1.3 nM T08922 CGM10E 72737641 IC50 = 8.2 nM T08922 C62TME 73292366 IC50 = 16 nM T08922 CG53HT 73292549 IC50 = 4.5 nM T08922 C4V8WZ 73292552 IC50 = 10 nM T08922 C1Q6MP 73292553 IC50 = 19 nM T08922 C4IJ3R 73292554 IC50 = 6.7 nM T08922 CI3EB7 73292555 IC50 = 5 nM T08922 CPT40G 73292726 IC50 = 4.2 nM T08922 CS8CG7 73292728 IC50 = 1.7 nM T08922 CXB8C3 73350749 IC50 = 2600 nM T08922 CNL1F6 76310321 IC50 = 231 nM T08922 CGX0J8 76310322 IC50 > 10000 nM T08922 CMS6N3 76310323 IC50 = 178 nM T08922 CK23BH 76313993 IC50 = 355 nM T08922 C9TD1F 76317535 IC50 = 246 nM T08922 CQ5S4U 76317536 IC50 = 64 nM T08922 C8QFN0 76321259 IC50 = 335 nM T08922 CW0L4N 76321260 IC50 = 166 nM T08922 CYC65M 76321261 IC50 = 244 nM T08922 CQ1F4P 76321262 IC50 = 128 nM T08922 C6XVJ2 76321263 IC50 = 2580 nM T08922 CJ32LQ 76324881 IC50 = 227 nM T08922 CX1G9D 76324882 IC50 = 103 nM T08922 C8GWZ7 76328439 IC50 = 486 nM T08922 CWB7L2 76328440 IC50 = 39 nM T08922 CJ41GZ 76328441 IC50 = 258 nM T08922 CRL3Y0 76328442 IC50 = 5.4 nM T08922 C36TCF 76328443 IC50 = 40 nM T08922 C84CZX 76332123 IC50 = 789 nM T08922 C4KSJ9 76332124 IC50 = 1830 nM T08922 C32YSB 76332125 IC50 = 159 nM T08922 CT0Z6Q 76335742 IC50 = 9.8 nM T08922 CKL9Y2 76335743 IC50 = 273 nM T08922 CM09JC 76335744 IC50 = 71 nM T08922 CFW1I2 78135022 IC50 = 60 nM T08922 CUAT74 89668981 IC50 = 180 nM T08922 CK1EP0 91936972 IC50 = 800 nM T08922 CMAP09 91936973 IC50 = 110 nM T08922 CPO08K 118344339 IC50 = 79 nM T08922 CTCQ02 118344344 IC50 = 6.9 nM T08922 C1HX3A 118344346 IC50 = 186 nM T08922 CI7P6J 118344348 IC50 = 46 nM T08922 C8J1PY 118344351 IC50 = 84 nM T08922 CAWZ16 118344383 IC50 = 48 nM T08922 CSUK24 118344385 IC50 = 306 nM T08922 CA1YM6 118344504 IC50 = 76 nM T08922 CC3N6Z 118344616 IC50 = 454 nM T08922 CC0RD7 118345442 IC50 = 26 nM T08922 CK43EA 118345549 IC50 = 4.3 nM T08922 C0MCW3 118346170 IC50 = 473 nM T08922 C0ORU1 118723380 IC50 = 78 nM T08922 CXIC05 118723381 IC50 = 1100 nM T08922 C4QX2V 118723382 IC50 = 161 nM T08922 CCG19A 118730172 IC50 = 80 nM T08922 CJ9R6H 118730173 IC50 = 50 nM T08922 CP04UJ 122194516 IC50 = 2200 nM T08922 C9J2QG 122194517 IC50 = 1000 nM T08922 CA85YT 122194518 IC50 = 2400 nM T08922 CI82JO 122194519 IC50 = 20000 nM T08922 CN7F5Q 122194520 IC50 > 10000 nM T08922 C8ZEU4 122194521 IC50 = 1400 nM T08922 CK28TA 122194522 IC50 = 880 nM T08922 C8HL0P 122194523 IC50 = 4500 nM T08922 CK8UF6 122194524 IC50 = 800 nM T08922 CXOM47 122194525 IC50 = 4000 nM T08922 C7HSC0 122194526 IC50 = 260 nM T08922 CGTE47 122194527 IC50 = 9200 nM T08922 CX9SO6 122194528 IC50 = 900 nM T08922 C4W8CM 122194529 IC50 > 14000 nM T08922 C6IJB7 122194530 IC50 = 5500 nM T08922 CS5L2D 122194531 IC50 = 1100 nM T08922 C1AV9M 122194532 IC50 = 200 nM T08922 CM1S7B 122370046 IC50 = 290 nM T08922 C2ULR6 130472593 IC50 = 1400 nM T08922 C56RIT 130472602 IC50 > 10000 nM T08922 CM91PV 130472623 IC50 = 5800 nM T08922 CPC2W5 130472637 IC50 > 10000 nM T08922 CG7ZR0 130472643 IC50 > 10000 nM T08922 C8QRE9 130472655 IC50 = 140 nM T08922 CK8TD2 130472676 IC50 = 77 nM T08922 CSHK51 130472735 IC50 > 10000 nM T08922 CJ48IH 130472776 IC50 > 10000 nM T08922 C19KAY 130472798 IC50 > 10000 nM T08922 C90QJL 130472810 IC50 = 170 nM T08922 CB2OR1 130472825 IC50 = 80 nM T08922 C4XMP1 130472850 IC50 > 10000 nM T08922 CN78SE 132578433 IC50 = 16 nM T08922 C36ESP 132578434 IC50 = 220 nM T08922 CR9CH0 134132369 IC50 = 48 nM T08922 CC3P5W 134135268 IC50 = 100 nM T08922 C1HYS8 134137111 IC50 = 260 nM T08922 CSGN69 134138458 IC50 = 1100 nM T08922 CX69BS 134139597 IC50 = 420 nM T08922 C6MVF5 134145715 IC50 = 7500 nM T08922 CVF58Q 134149423 IC50 = 610 nM T08922 CB06NG 134226781 IC50 = 95 nM T08922 C0NEF2 134226787 IC50 > 10000 nM T08922 C3PXH5 134226791 IC50 = 860 nM T08922 C2XVM6 134226798 IC50 > 10000 nM T08922 CQF87J 134226821 IC50 = 930 nM T08922 CSEL43 134226826 IC50 = 5700 nM T08922 C13UJI 134226866 IC50 = 290 nM T08922 CV69CF 136164076 IC50 = 0.21 nM T08922 CC0QA2 145967606 IC50 = 1.9 nM T08922 C19IVD 145967885 IC50 = 59 nM T08922 C2S8DE 145969909 IC50 = 66 nM T08922 CI3O2K 145970611 IC50 = 25 nM T08922 C6CD4Z 145970793 IC50 = 10 nM T08922 CS5U3M 145970807 IC50 = 253 nM T08922 C68MEO 145982863 IC50 = 944 nM T08922 C0UK4O 145983273 IC50 > 5000 nM T08922 CWC6X7 145983307 IC50 = 3021 nM T08922 C93NVW 145983529 IC50 > 5000 nM T08922 CIY63H 145983729 IC50 = 764 nM T08922 CE6Q3M 145983942 IC50 = 2738 nM T08922 CMD9A2 145984050 IC50 = 1882 nM T08922 C30XCZ 145984055 IC50 = 397 nM T08922 CCM6V3 145984070 IC50 > 5000 nM T08922 CCIR92 145984514 IC50 > 5000 nM T08922 CWD59X 145984988 IC50 > 5000 nM T08922 CI83ZU 145985112 IC50 = 1237 nM T08922 C6H4QT 145985213 IC50 = 1112 nM T08922 CHO23R 145985261 IC50 > 5000 nM T08922 C5B3MJ 145985287 IC50 = 3772 nM T08922 C2KNC8 145985487 IC50 > 5000 nM T08922 C9LWB4 145985500 IC50 = 976 nM T08922 C9C2RK 145985542 IC50 = 3477 nM T08922 CXD73B 145986022 IC50 = 4646 nM T08922 C2DM5H 145986295 IC50 = 1944 nM T08922 C7O1PF 145987480 IC50 = 40 nM T08922 C81LEH 145987485 IC50 = 2.1 nM T08922 C6B8VZ 155524377 IC50 = 3700 nM T08922 C7K5IL 155526152 IC50 = 2200 nM T08922 CE0FM4 155566710 IC50 = 6400 nM T08922 CJ23QI 155566749 IC50 = 2000 nM T08922 C7Q3XR 155567174 IC50 = 4000 nM T08922 D07WIC 449097 IC50 = 34 nM T08922 D0IY5Y 11675600 IC50 = 75 nM T17852 D05MQK 110635 IC50 > 10000 nM T17852 D0C9SY 135400189 IC50 = 460 nM T17852 D0Z7ZM 135398744 IC50 = 3600 nM T17852 D0A9IY 135564558 IC50 = 8.3 nM T17852 D0T5PO 5092 IC50 > 16000 nM T17852 D0W7UN 135908617 IC50 = 52 nM T17852 D0X0PP 59351313 IC50 > 30000 nM T17852 D05VBJ 71295299 IC50 > 10000 nM T17852 D0WS3T 72706254 IC50 > 10000 nM T17852 D00YPW 135399235 Ki = 35000 nM T17852 C1H8NR 155248 IC50 > 100000 nM T17852 CYWS98 185848 IC50 > 100000 nM T17852 C8JLO0 2243267 IC50 > 10000 nM T17852 CW42OS 2857518 IC50 = 8000 nM T17852 C45VZC 11438405 IC50 > 16000 nM T17852 C4ZYH9 11547485 IC50 > 10000 nM T17852 CUK49V 11988837 Ki = 6100 nM T17852 CFIO49 11988967 Ki > 100000 nM T17852 C2D0NG 11989101 Ki = 50000 nM T17852 C65ABT 11989102 Ki > 100000 nM T17852 C1B4XD 11992634 IC50 > 2000 nM T17852 CPX16N 11993169 IC50 > 2000 nM T17852 C1PZ8C 18734933 IC50 > 16000 nM T17852 CW96SI 23624262 IC50 > 1000 nM T17852 C4S6VD 23654252 IC50 > 50000 nM T17852 C9WGI4 24802717 IC50 > 5000 nM T17852 C93DZI 25147798 IC50 > 50000 nM T17852 CPC08B 25179287 IC50 > 50000 nM T17852 COB03R 25179478 IC50 > 50000 nM T17852 CICF39 42629702 IC50 > 10000 nM T17852 CM3X9S 42629827 IC50 > 1000 nM T17852 CQN26J 42629945 IC50 > 1000 nM T17852 C6O5FX 42630062 IC50 > 10000 nM T17852 C71ZNR 42630180 IC50 > 10000 nM T17852 C4RHY0 42630191 IC50 > 10000 nM T17852 CT6RS9 42630192 IC50 > 10000 nM T17852 CYZL43 42630317 IC50 > 10000 nM T17852 CH42OZ 42630318 IC50 > 10000 nM T17852 C7X5AH 42630437 IC50 > 10000 nM T17852 CW8OB3 44243146 Ki > 10000 nM T17852 C5IMB2 46239424 Ki > 10000 nM T17852 CKR9P7 46239425 Ki > 10000 nM T17852 CI1F5C 46239840 Ki >= 770 nM T17852 C26XVS 46240044 Ki >= 4793 nM T17852 CE4JU7 46842025 IC50 > 10000 nM T17852 CR8JC2 46842169 IC50 > 10000 nM T17852 CC4EI5 46881198 IC50 = 103 nM T17852 CPQ69R 46881199 IC50 = 22 nM T17852 C3P2IN 46933992 IC50 >= 55000 nM T17852 CHA5Z0 49821469 IC50 > 1000 nM T17852 C1AYP0 49821627 IC50 > 500 nM T17852 C85AXR 49821714 IC50 > 1000 nM T17852 CZS03D 50902030 Ki > 4274 nM T17852 CH2Z1E 50902289 Ki > 7100 nM T17852 C4HJL2 50902291 Ki > 7950 nM T17852 C6A1IU 50902549 Ki > 2000 nM T17852 C3Y2AV 50903255 Ki > 2000 nM T17852 CGF65A 54670110 IC50 > 30000 nM T17852 C90ZLC 54670399 IC50 > 30000 nM T17852 C4TGL7 56648496 IC50 > 1000 nM T17852 CH6C3L 56648679 IC50 > 10000 nM T17852 CCY79V 56648680 IC50 > 10000 nM T17852 CNE96P 56648857 IC50 > 10000 nM T17852 CX86AQ 56648859 IC50 > 5000 nM T17852 CPC3T4 56654131 IC50 > 10000 nM T17852 C0YD3P 56928304 IC50 > 5000 nM T17852 C8RO6A 56929788 IC50 > 1000 nM T17852 CG3DF1 57392948 Ki > 10000 nM T17852 CE36TV 57394695 Ki > 10000 nM T17852 CPA3D1 57403394 Ki > 10000 nM T17852 C4XMB6 58547809 IC50 > 30000 nM T17852 CEB3G9 58547814 IC50 > 30000 nM T17852 C08QVG 58547833 IC50 > 30000 nM T17852 CFVG67 58547863 IC50 > 30000 nM T17852 CYZA38 58548077 IC50 > 30000 nM T17852 CY8J3O 68181896 IC50 > 10000 nM T17852 CC43LF 71074083 IC50 > 10000 nM T17852 C4P0XT 71092344 IC50 > 30000 nM T17852 C6DAG4 71092519 IC50 > 30000 nM T17852 C2HGI7 71153408 IC50 > 10000 nM T17852 C9GR3L 71153436 IC50 > 10000 nM T17852 C4GNJ3 71598545 IC50 > 1000 nM T17852 C68SDB 71719394 IC50 > 10000 nM T17852 CZ0G2X 72165213 IC50 > 10000 nM T17852 C7XRY6 72190879 IC50 > 30000 nM T17852 CQ3GD7 72704434 Ki = 17000 nM T17852 C9JE6M 75815419 IC50 > 200 nM T17852 CF03DW 90168772 IC50 > 20000 nM T17852 CM6J9K 90168778 IC50 > 20000 nM T17852 C1JPD6 91844700 IC50 > 10000 nM T17852 C7F6JY 92135987 IC50 > 10000 nM T17852 CYQV05 92471958 IC50 = 350 nM T17852 C0YZ1T 101893663 IC50 = 15000 nM T17852 CSED17 101893664 IC50 = 8800 nM T17852 CSCY01 117949009 IC50 > 10000 nM T17852 CYQ74R 118479645 IC50 > 10000 nM T17852 CQ9X2T 118525749 IC50 > 10000 nM T17852 CA9Z4N 118525753 IC50 > 10000 nM T17852 COM19L 118525755 IC50 > 10000 nM T17852 CCB0S9 118525772 IC50 > 10000 nM T17852 C0SV3H 118525773 IC50 > 10000 nM T17852 CG4Z8E 118525774 IC50 > 10000 nM T17852 CYE6W5 118525795 IC50 > 10000 nM T17852 C8OH0Y 118525801 IC50 > 10000 nM T17852 CP75JF 118525805 IC50 > 10000 nM T17852 CR65SL 118525810 IC50 > 10000 nM T17852 C94ZTQ 118525830 IC50 > 10000 nM T17852 CM8IQ7 118525835 IC50 > 10000 nM T17852 CQ0LU1 118525854 IC50 > 10000 nM T17852 C2PWK5 118534656 IC50 > 10000 nM T17852 C4H2LG 118534683 IC50 > 10000 nM T17852 CVYK24 118556943 IC50 > 50000 nM T17852 CMZC83 118720798 IC50 = 10100 nM T17852 C7YE2L 118720799 IC50 = 5600 nM T17852 C20SPH 118720800 IC50 = 6400 nM T17852 C6DQK7 118720801 IC50 = 7700 nM T17852 C4RZB1 118720802 IC50 = 7800 nM T17852 C4CLB3 118720803 IC50 = 6700 nM T17852 CRJE23 122185011 IC50 > 30000 nM T17852 CS6M9C 122193679 IC50 > 100000 nM T17852 CVX7U9 127029185 IC50 = 4830 nM T17852 C4UR7D 127038167 IC50 > 1000 nM T17852 C4H2TJ 127038168 IC50 > 1000 nM T17852 CL9JT8 127038169 IC50 > 1000 nM T17852 CJPX60 127038509 IC50 > 1000 nM T17852 C26EAG 127038511 IC50 > 1000 nM T17852 CTM9E4 127038512 IC50 > 1000 nM T17852 C6AQ2U 127038513 IC50 > 1000 nM T17852 CV1FM0 127038868 IC50 > 1000 nM T17852 CADU23 127038869 IC50 > 1000 nM T17852 C62CSI 129051756 IC50 > 10000 nM T17852 C5RFV2 129051760 IC50 > 10000 nM T17852 CH20AQ 129051764 IC50 > 10000 nM T17852 CDJ2V1 129051781 IC50 > 10000 nM T17852 C7AD3Z 129051788 IC50 > 10000 nM T17852 CACJ46 132489333 IC50 > 10000 nM T17852 C2P1IU 134129996 IC50 > 100000 nM T17852 CLE03O 134130328 IC50 > 100000 nM T17852 CSN6J0 134130563 IC50 > 100000 nM T17852 C0A1CZ 134131162 IC50 > 100000 nM T17852 CZ09EG 135418212 IC50 = 10 nM T17852 C7GC0D 135436665 IC50 = 36 nM T17852 C1RD6B 135443112 IC50 = 2100 nM T17852 C3R8SE 135457869 IC50 = 41 nM T17852 CWQG94 135484473 IC50 = 56 nM T17852 C2E3GU 135541419 IC50 = 22 nM T17852 CW51OH 135566500 IC50 = 0.8 nM T17852 CR8JM9 135566501 IC50 = 66 nM T17852 CN87GS 135566743 IC50 = 11 nM T17852 CYVU41 135566744 IC50 = 32 nM T17852 CHDC83 135566745 IC50 > 10000 nM T17852 C9IJK1 135566935 IC50 = 0.6 nM T17852 CX7I5Z 135721222 IC50 = 82 nM T17852 CL34KC 135860085 IC50 = 150 nM T17852 CU1W4H 135860086 IC50 = 38.02 nM T17852 C9FO2W 135860090 IC50 = 194.98 nM T17852 CH5N1M 135860091 IC50 = 28.84 nM T17852 C13QRM 135860092 IC50 = 16 nM T17852 CHT23I 135860093 IC50 = 10.96 nM T17852 C38XKR 135860094 IC50 = 10.72 nM T17852 C26ECA 135860095 IC50 = 12.3 nM T17852 CLM59K 135860101 IC50 = 1.9 nM T17852 C7QAS6 135873861 IC50 = 22 nM T17852 CWYC37 135873891 IC50 = 47 nM T17852 CI31NQ 135873914 IC50 = 230 nM T17852 CS9DT5 135875901 IC50 = 63 nM T17852 CPM68I 135875902 IC50 = 11 nM T17852 C87UJS 135875904 IC50 = 14.79 nM T17852 CVZ12B 135886459 IC50 = 4.9 nM T17852 CCH2Z5 135886460 IC50 = 4.6 nM T17852 CVP62I 135886467 IC50 = 3.8 nM T17852 CA53FG 135886468 IC50 = 12 nM T17852 C6T1EH 135886483 IC50 = 1.2 nM T17852 C0HJ2E 135886489 IC50 = 0.9 nM T17852 C09WPF 135886491 IC50 = 1.7 nM T17852 C3E7IT 135886495 IC50 = 4.6 nM T17852 C8Q7TD 135886496 IC50 = 3.4 nM T17852 CTX54Z 135896326 IC50 = 35 nM T17852 CRP84K 135908600 IC50 = 1 nM T17852 CH6QL0 136059722 IC50 = 530 nM T17852 C2J7ZU 136059723 IC50 = 87 nM T17852 CN06GO 136059724 IC50 = 19 nM T17852 C8EA6G 136059725 IC50 = 46 nM T17852 C31KAG 136059726 IC50 = 23 nM T17852 C12UMG 136059728 IC50 = 7 nM T17852 C1CIB0 136079019 IC50 = 7470 nM T17852 CAF6W1 136079038 IC50 = 7510 nM T17852 CGPB91 136087043 IC50 = 52 nM T17852 CWMC50 136087044 IC50 = 5.5 nM T17852 CRP24A 136087045 IC50 = 3 nM T17852 CA7B3X 136087046 IC50 = 8.1 nM T17852 C32NKJ 136087047 IC50 = 25.9 nM T17852 C4EGK9 136087048 IC50 = 1.05 nM T17852 CU5DG1 136087049 IC50 = 17.6 nM T17852 C7SUX4 136087050 IC50 = 6.4 nM T17852 CU9JX5 136087051 IC50 = 1.1 nM T17852 CAH15U 136128521 IC50 = 6.3 nM T17852 CW2AZ7 136128560 IC50 = 89 nM T17852 C21FVA 136180322 IC50 = 3800 nM T17852 CQW7T0 136197286 IC50 > 10000 nM T17852 C58DCK 136217453 IC50 = 721 nM T17852 CI96YZ 136217454 IC50 = 52 nM T17852 C8TQ7A 136217455 IC50 = 21 nM T17852 CJK71T 136217456 IC50 = 696 nM T17852 C1MQ5T 136217457 IC50 = 595 nM T17852 C4G8LD 136217458 IC50 = 237 nM T17852 CI0X1E 136217463 IC50 = 308 nM T17852 C8PQZ1 136217464 IC50 = 204 nM T17852 CBQ31P 136236301 IC50 = 152 nM T17852 CJ47RH 136236303 IC50 = 148 nM T17852 CR36FZ 136236304 IC50 > 1000 nM T17852 C8RZ2L 136236305 IC50 > 1000 nM T17852 C29SJC 136236306 IC50 = 593 nM T17852 CB06CO 136236307 IC50 > 1000 nM T17852 CL20MP 136236308 IC50 > 1000 nM T17852 CRV5F8 136236309 IC50 = 986 nM T17852 C27HTA 136236310 IC50 = 7 nM T17852 CI17ZJ 136236311 IC50 = 19 nM T17852 CCWE64 136236312 IC50 = 43 nM T17852 CDY5T0 136236313 IC50 = 70 nM T17852 C9K7JN 136236314 IC50 = 64 nM T17852 C5JGW8 136236315 IC50 = 57 nM T17852 CI6R9B 136236316 IC50 = 50 nM T17852 C15POR 136242452 IC50 = 63 nM T17852 C2C7YL 136242453 IC50 = 45 nM T17852 CRPN39 136645466 IC50 > 10000 nM T17852 CLE62X 137179301 IC50 > 10000 nM T17852 C54KGS 137300710 IC50 = 4800 nM T17852 C2N9VT 137348687 IC50 > 10000 nM T17852 C6KYD7 137700754 IC50 = 8.7 nM T17852 CM3UF7 137700779 IC50 > 20000 nM T17852 CPTE92 138319693 IC50 > 32000 nM T17852 C2QLX3 138393292 IC50 > 50000 nM T17852 CMW20N 141737696 IC50 > 4000 nM T17852 C8HEG7 141737705 IC50 > 3000 nM T17852 C70YLA 145953136 IC50 > 10000 nM T17852 C0C6FG 145954733 IC50 > 10000 nM T17852 CH7VB3 145957961 IC50 > 10000 nM T17852 C3IU8W 145965666 IC50 = 55 nM T17852 C0DYA1 145967207 IC50 = 16 nM T17852 CL36HK 145967227 IC50 = 899 nM T17852 CC7HN2 145974174 IC50 > 100000 nM T17852 CK1BR0 145978345 IC50 > 100000 nM T17852 CT83WZ 145982175 IC50 = 65 nM T17852 C6P5GN 145982663 IC50 = 2.8 nM T17852 CA6IP4 145983673 IC50 = 850 nM T17852 C1JB4T 145983923 IC50 = 750 nM T17852 C9M4GK 145989574 IC50 = 590 nM T17852 C7LN8Q 145989614 IC50 = 200 nM T17852 CD7HJ8 145990073 IC50 = 220 nM T17852 CE7Z5R 145991006 IC50 = 180 nM T17852 CO4PB7 145991254 IC50 = 210 nM T17852 CHJ79V 145997874 IC50 > 10000 nM T17852 CM7TX2 148279038 IC50 > 100000 nM T17852 CADM48 155510637 IC50 = 112 nM T17852 CT5EQ7 155511060 IC50 = 103 nM T17852 CV0Y5H 155512206 IC50 = 24 nM T17852 CHPM03 155517492 IC50 = 100 nM T17852 CGLS24 155521088 IC50 = 20 nM T17852 CL8CU6 155521936 IC50 > 200000 nM T17852 CYI51O 155523485 IC50 = 594 nM T17852 C9CYA3 155525884 IC50 = 91 nM T17852 CT85RG 155530589 IC50 > 200000 nM T17852 CQ7IJ0 155531325 IC50 = 88 nM T17852 C07WDO 155532938 IC50 = 13 nM T17852 C0M2UC 155539455 IC50 = 15 nM T17852 C3KE9M 155548362 IC50 = 227 nM T17852 CQ5P0M 155553114 IC50 = 49 nM T17852 C35CKI 155554168 IC50 = 34000 nM T17852 CX6F2U 155559756 IC50 = 19 nM T17852 C2DA1W 155561694 IC50 = 13900 nM T17852 CQ2R0W 155568588 IC50 = 32300 nM T17852 D06NIT 135564899 IC50 = 1.778 nM T17852 D09RKU 46239428 Ki > 10000 nM T17852 D0R6MT 3758 IC50 > 117000 nM T17852 D0V4WB 149790 IC50 > 16000 nM T26203 D06WTZ 53232 IC50 = 8 ug.mL-1 T26203 D0Q9EV 11965427 IC50 = 2.98 nM T26203 CKM1X8 128677 IC50 = 140 nM T26203 CXI3Y4 645569 IC50 > 100000 nM T26203 C5Q0FP 745480 IC50 = 56000 nM T26203 CYBV18 916176 IC50 > 100000 nM T26203 C16YNJ 962611 IC50 = 99000 nM T26203 COB6U4 2807642 IC50 = 6300 nM T26203 CYBK67 5481003 IC50 = 4000 nM T26203 CF2B7X 6442405 IC50 > 50 ug.mL-1 T26203 CT3BF9 9797597 IC50 = 170 nM T26203 C74QCT 9798233 IC50 = 99 nM T26203 CCI90K 9799728 IC50 = 600 nM T26203 C18UGE 9818339 IC50 = 11000 nM T26203 CJQ2W6 9835897 IC50 > 1000 nM T26203 C6G5RT 9836507 IC50 > 4000 nM T26203 CUGN49 9836683 IC50 = 82 nM T26203 CJ5SU0 9839311 IC50 = 25 nM T26203 CSK6P4 9841875 IC50 = 1400 nM T26203 CJ6K2V 9847995 IC50 = 63 nM T26203 C5DRX6 9856682 IC50 = 120 nM T26203 C9MA3Z 9858009 IC50 = 16 nM T26203 C0ZQV7 9858022 IC50 = 54 nM T26203 C3MG0X 9860649 IC50 = 1900 nM T26203 C8IO4M 9878726 IC50 = 92000 nM T26203 C91VCO 9878930 IC50 = 20 nM T26203 CP34JF 9879093 IC50 = 570 nM T26203 C5S6CZ 9879529 IC50 = 9 nM T26203 CBKH73 9880710 IC50 = 180 nM T26203 C1L5WE 9880711 IC50 = 34 nM T26203 C0O5BM 9881984 IC50 = 3600 nM T26203 C0W1SB 9882382 IC50 = 2300 nM T26203 CY7KG3 9883504 IC50 = 10 nM T26203 CL1FR4 9900816 IC50 = 2 nM T26203 C3D1XN 9900943 IC50 = 430 nM T26203 C9DHR2 9901085 IC50 = 770 nM T26203 CRND31 9901574 IC50 = 150 nM T26203 CBM7Y3 9903965 IC50 = 2300 nM T26203 CKJ7T0 9903998 IC50 = 6600 nM T26203 C1JI7S 9904207 IC50 = 5000 nM T26203 C3VJ9K 9904395 IC50 = 250 nM T26203 C62JUP 9904430 IC50 > 4000 nM T26203 CYN51E 9905179 IC50 = 48 nM T26203 CDML85 9906347 IC50 = 3 nM T26203 CO63ID 9921367 IC50 = 1800 nM T26203 CQ4WG3 9921987 IC50 = 160 nM T26203 C9T3ME 9922373 IC50 = 140 nM T26203 CO5L2R 9922793 IC50 = 47 nM T26203 C36KVQ 9922943 IC50 = 160 nM T26203 CW5P9J 9924766 IC50 = 37 nM T26203 CYKV73 9934394 IC50 = 240 nM T26203 CB85IM 9935010 IC50 = 700 nM T26203 C7QP1H 9944101 IC50 = 20 nM T26203 C2JZW5 9944163 IC50 = 40 nM T26203 C9AJP0 9944774 IC50 = 140 nM T26203 CL9I6U 9945784 IC50 = 13 nM T26203 CB3P7T 9946091 IC50 > 1000 nM T26203 CYJ59B 9946991 IC50 = 25 nM T26203 CAFK13 9947244 IC50 = 10 nM T26203 CR4LP3 9948282 IC50 = 39000 nM T26203 CNH47D 9948311 IC50 = 3700 nM T26203 C0YEQ7 9952465 IC50 = 75 nM T26203 C2TYQ1 9953413 IC50 > 100000 nM T26203 CBD1W8 9954095 IC50 = 2100 nM T26203 CKH98V 9957380 IC50 = 140 nM T26203 CWH3L0 9965679 IC50 = 25 nM T26203 CI4DU5 9966679 IC50 = 32 nM T26203 CFEI36 9967126 IC50 = 110 nM T26203 CA5W9Z 9967290 IC50 = 680 nM T26203 CS9DM3 9967511 IC50 = 690 nM T26203 CYXW91 9968489 IC50 = 39 nM T26203 CVNR86 9979502 IC50 = 270 nM T26203 CUZI90 10019432 IC50 = 5900 nM T26203 CSD14A 10054168 IC50 = 360 nM T26203 C1RUK3 10070771 IC50 = 270 nM T26203 CX30HT 10089338 IC50 = 1 nM T26203 CT0Y2E 10097459 IC50 = 190 nM T26203 C4E8NU 10106199 IC50 = 3500 nM T26203 COIF97 10107659 IC50 = 6600 nM T26203 CY23GM 10108997 IC50 = 1400 nM T26203 C2P4UO 10110987 IC50 > 4000 nM T26203 CTW3P9 10116693 IC50 = 26 nM T26203 C07COW 10132518 IC50 = 110 nM T26203 C6N1FU 10134148 IC50 > 4000 nM T26203 CH49BD 10154440 IC50 = 680 nM T26203 COF2S9 10154441 IC50 = 18 nM T26203 CL7H2B 10154801 IC50 = 340 nM T26203 C0CP1T 10155661 IC50 = 320 nM T26203 CSB5F9 10156828 IC50 = 300 nM T26203 CF4DP2 10177047 IC50 = 53 nM T26203 C6RN4F 10178848 IC50 = 4 nM T26203 CHN3X1 10202790 IC50 > 4000 nM T26203 CD95KA 10221525 IC50 = 490 nM T26203 C23UCO 10252638 IC50 = 100 nM T26203 CJZU30 10267771 IC50 = 8 nM T26203 C2OQ0K 10267925 IC50 = 580 nM T26203 C9C0UG 10291112 IC50 > 4000 nM T26203 CWZU32 10291698 IC50 = 46 nM T26203 CTUP45 10291904 IC50 > 4000 nM T26203 CM05NG 10298900 IC50 = 130 nM T26203 C7KO6U 10361323 IC50 = 5 nM T26203 C1NX9Z 10469899 IC50 < 30000 nM T26203 CZ3DK8 10566084 IC50 = 19000 nM T26203 C5Q8EF 10566766 IC50 = 12000 nM T26203 CN3H5M 10632359 IC50 = 360 nM T26203 C6QZG3 10686899 IC50 > 4000 nM T26203 CZF1H3 10708446 IC50 = 540 nM T26203 CAPG02 10732433 IC50 = 840 nM T26203 CKJS90 10739377 IC50 = 5300 nM T26203 C6K5GC 10860379 IC50 = 40 nM T26203 C7CL4Z 10860782 IC50 = 270 nM T26203 CSO95L 10862219 IC50 > 901 nM T26203 C7OFZ9 10863087 IC50 = 120 nM T26203 C5PWJ4 10874238 IC50 = 270 nM T26203 C6PRJ8 10880644 IC50 = 42 nM T26203 CV9I3D 10891751 IC50 = 2 nM T26203 C9X6VP 10892285 IC50 = 780 nM T26203 C9DUB8 10892642 IC50 = 10 nM T26203 CS1T3C 10896625 IC50 = 116 nM T26203 CARC06 10904579 IC50 = 360 nM T26203 CHWL69 10905666 IC50 = 16 nM T26203 CZ9N5L 10906388 IC50 = 270 nM T26203 CLPA31 10906508 IC50 = 32 nM T26203 CNO84S 10906650 IC50 = 270 nM T26203 C7YG6L 10924566 IC50 = 23 nM T26203 C2XU9N 10928517 IC50 = 270 nM T26203 CFA83X 10957497 IC50 = 270 nM T26203 C5UR1K 10960480 IC50 = 270 nM T26203 CY2OD3 10960504 IC50 = 270 nM T26203 CR51AV 10970154 IC50 = 4 nM T26203 CQ6E7Y 10970207 IC50 > 1000 nM T26203 CB31OE 10980658 IC50 = 760 nM T26203 C32YBT 10980772 IC50 = 270 nM T26203 C94UAC 10982608 IC50 = 5 nM T26203 CP51XQ 10992466 IC50 = 270 nM T26203 C67HEX 10992857 IC50 = 270 nM T26203 CQ2LN7 11001466 IC50 = 270 nM T26203 CVR4Y3 11001541 IC50 = 31 nM T26203 CG8R2I 11002350 IC50 = 270 nM T26203 CCP7K5 11013542 IC50 = 5 nM T26203 C1ZRL6 11014018 IC50 = 6 nM T26203 CIW6J5 11023935 IC50 = 17 nM T26203 C7NCE4 11036406 IC50 = 1.4 nM T26203 CM5HI8 11045962 IC50 = 5 nM T26203 C7U2JK 11048059 IC50 = 22 nM T26203 C7E6GN 11048585 IC50 = 670 nM T26203 CNHY70 11057712 IC50 = 79 nM T26203 COE6W0 11068095 IC50 = 6 nM T26203 C9Q0MP 11070710 IC50 = 820 nM T26203 CHT7C5 11076507 IC50 = 270 nM T26203 CZSV01 11078679 IC50 > 970 nM T26203 C1KE2T 11079237 IC50 = 8 nM T26203 C06TWP 11080019 IC50 = 270 nM T26203 C8SRX4 11080157 IC50 = 790 nM T26203 CT0I6A 11088702 IC50 = 270 nM T26203 C5T1BO 11089640 IC50 = 6 nM T26203 C3MO4P 11090180 IC50 = 270 nM T26203 CQYV18 11091464 IC50 = 730 nM T26203 CPM54S 11100349 IC50 = 270 nM T26203 CSF94U 11102008 IC50 = 580 nM T26203 C51PTF 11109642 IC50 = 18 nM T26203 C8RF0J 11111846 IC50 > 1000 nM T26203 C8WI4X 11120977 IC50 = 150 nM T26203 CUGV75 11122788 IC50 > 1000 nM T26203 CHIT70 11134430 IC50 = 53 nM T26203 CRPC48 11134652 IC50 = 600 nM T26203 CA20RU 11187409 IC50 = 530 nM T26203 CFGJ28 11200368 IC50 = 420 nM T26203 CJ1NO9 11200918 IC50 = 420 nM T26203 CIU31Z 11235306 IC50 = 420 nM T26203 C5WRM2 11315070 IC50 = 420 nM T26203 CY57WM 11326937 IC50 = 420 nM T26203 C7H8BD 11428675 IC50 = 470 nM T26203 C4HYP3 11429387 IC50 = 420 nM T26203 C45CZE 11741193 IC50 = 270 nM T26203 C5DUF4 11760748 IC50 = 120 nM T26203 CG60JO 11772244 IC50 = 420 nM T26203 CF7GU9 11777631 IC50 < 30000 nM T26203 C8BJ0L 11783098 IC50 = 160 nM T26203 C43LZD 11783922 IC50 = 830 nM T26203 CKRM28 11793014 IC50 > 1000 nM T26203 CLX8Z9 11825588 IC50 = 4 nM T26203 C7SG8X 11828434 IC50 = 3.8 nM T26203 C6PWB3 16041827 IC50 = 30 ug.mL-1 T26203 CC83DL 16098225 IC50 = 10.7 ug.mL-1 T26203 C2A0PI 18670114 IC50 = 3000 nM T26203 CUW59L 23564498 IC50 = 420 nM T26203 CZ0U6W 25255091 IC50 > 50 ug.mL-1 T26203 C36WMA 44264201 IC50 > 4000 nM T26203 CM7P9U 44344139 IC50 = 59 nM T26203 CJ14IR 145957451 IC50 = 420 nM T26203 D03YAG 21580213 IC50 = 13.4 ug.mL-1 T26203 D07XCA 9846729 IC50 = 35 nM T26203 D0H0FG 6439947 IC50 = 6 ug.mL-1 T26203 D0S2UZ 9974595 IC50 = 8.8 ug.mL-1 T26203 D0ZH9W 5318516 IC50 = 13.5 ug.mL-1 T05089 C8KY3N 867752 IC50 > 20000 nM T05089 CG0L5Q 1107220 IC50 = 130 nM T05089 C9M6AJ 1107221 IC50 = 260 nM T05089 CC05UR 1107239 IC50 = 1300 nM T05089 C6R5UW 1268403 IC50 = 660 nM T05089 CT2WE8 1356077 IC50 > 20000 nM T05089 C5JL9Z 2898877 IC50 = 2100 nM T05089 CTS84G 3368574 IC50 = 5000 nM T05089 C8R4MK 3657956 IC50 = 3000 nM T05089 CSI6B2 3727899 IC50 > 10000 nM T05089 C1MQ6J 3825946 IC50 = 170 nM T05089 CAZM48 4248009 IC50 = 1200 nM T05089 C3PIJ1 4257218 IC50 > 20000 nM T05089 C5X2LP 6870687 IC50 = 890 nM T05089 CTQ4X2 9556542 IC50 = 97 nM T05089 C1WAS7 9557280 IC50 = 25700 nM T05089 C7K9NM 9557402 IC50 > 100000 nM T05089 CUMP58 9642456 IC50 = 31300 nM T05089 CHW90Z 9651715 IC50 = 210 nM T05089 CDY4V7 9652824 IC50 > 100000 nM T05089 CEFS86 11518047 IC50 = 5000 nM T05089 CW5ZH3 32887072 IC50 > 100000 nM T05089 CEV6S1 49959483 IC50 = 19400 nM T05089 CFK48S 49959506 IC50 = 63800 nM T05089 CT4KN6 70681931 IC50 = 5900 nM T05089 CH2UD8 70681941 IC50 = 23500 nM T05089 CN45QJ 70681942 IC50 = 13300 nM T05089 C95YFT 70681943 IC50 = 6300 nM T05089 CJ2L0P 70684057 IC50 = 23000 nM T05089 CUE20O 70684058 IC50 = 10400 nM T05089 CDN5V6 70684059 IC50 = 3200 nM T05089 CF3I8R 70686195 IC50 = 11200 nM T05089 C0WDI6 70686196 IC50 = 10800 nM T05089 CR2AG0 70686197 IC50 = 3300 nM T05089 C9NTX0 70686198 IC50 = 13100 nM T05089 CRQ71U 70686199 IC50 = 4900 nM T05089 CTFL70 70686200 IC50 = 2800 nM T05089 C26XDG 70688323 IC50 = 28700 nM T05089 CZ17CF 70688327 IC50 = 25900 nM T05089 CQR14B 70688328 IC50 = 9000 nM T05089 C8NE6X 70690338 IC50 = 17300 nM T05089 CL7O8C 70690339 IC50 = 7700 nM T05089 C9APV5 70690340 IC50 = 3200 nM T05089 CUMI58 70690341 IC50 = 5200 nM T05089 CKB06C 70692505 IC50 = 27000 nM T05089 CMW51K 70694539 IC50 = 16300 nM T05089 CJ09KP 70694549 IC50 = 29200 nM T05089 C6WFC1 70694550 IC50 = 21200 nM T05089 CKAD56 70694551 IC50 = 15600 nM T05089 CYXV78 70694552 IC50 = 16300 nM T05089 C6KNH0 70694553 IC50 = 3800 nM T05089 CRT84S 70694554 IC50 = 26900 nM T05089 CV42YB 70696604 IC50 = 12300 nM T05089 CIW5X9 72165188 IC50 = 80 nM T05089 COV32B 110655853 IC50 > 100000 nM T05089 C2BD4F 126029515 IC50 > 100000 nM T05089 CWE3L1 126118288 IC50 = 370 nM T05089 CPM71Y 126120777 IC50 = 220 nM T05089 C94LTC 129897070 IC50 = 30 nM T05089 C87XQN 135362888 IC50 = 5000 nM T05089 CLMV79 135362963 IC50 = 230 nM T05089 CB4E2I 135362967 IC50 = 1300 nM T05089 CL2K6B 135362968 IC50 > 20000 nM T05089 CJEA01 135362969 IC50 = 2500 nM T05089 C7NOS2 135362985 IC50 > 20000 nM T05089 C0ECF1 135363016 IC50 = 1600 nM T05089 C7NBJ6 135363020 IC50 = 3000 nM T05089 CP61HB 135363040 IC50 = 380 nM T05089 CCR6Q4 135363059 IC50 = 180 nM T05089 C1VDL7 135363062 IC50 = 6200 nM T05089 CAP47J 135363284 IC50 = 2500 nM T05089 CZ9B6W 135363371 IC50 = 600 nM T05089 C79HRK 135460621 IC50 = 1000 nM T05089 CKY61A 137632563 IC50 = 1880 nM T05089 C48GVD 137633189 IC50 = 840 nM T05089 CNLH04 137634955 IC50 = 2700 nM T05089 CVKN20 137635893 IC50 > 20000 nM T05089 C0ZO5P 137636824 IC50 > 20000 nM T05089 CB74EV 137636987 IC50 = 1300 nM T05089 CEN35H 137639154 IC50 = 1300 nM T05089 C3L4RJ 137641611 IC50 > 20000 nM T05089 CF89YJ 137642052 IC50 = 450 nM T05089 C8WOE4 137645920 IC50 = 490 nM T05089 C4E3ZC 137650594 IC50 > 20000 nM T05089 CCQD85 137652022 IC50 = 230 nM T05089 C5N6AY 137653190 IC50 = 370 nM T05089 CH9LP7 137654007 IC50 = 3800 nM T05089 C2ZPX0 137655505 IC50 = 700 nM T05089 CT5Q3H 137655791 IC50 = 1300 nM T05089 C31DPR 137658006 IC50 = 150 nM T05089 C7LE9S 137658181 IC50 = 1300 nM T05089 C9Z2JE 137658371 IC50 = 925 nM T05089 C8JA5B 137660924 IC50 = 320 nM T05089 CX7N9O 147373071 IC50 > 100000 nM T05089 CU2NM3 148137406 IC50 = 21200 nM T05089 C4Y6EL 148455436 IC50 = 10700 nM T05089 C2BY7J 148848233 IC50 > 100000 nM T05089 CUXO84 153465084 IC50 > 100000 nM T05089 CDS7U0 153465085 IC50 > 100000 nM T05089 CMK62T 153465088 IC50 > 100000 nM T05089 CU25NA 153465089 IC50 = 15700 nM T05089 CA17VQ 153465091 IC50 = 22 nM T05089 C6YQ3A 153465093 IC50 = 300 nM T05089 CQ8G2P 153465094 IC50 > 100000 nM T05089 C0E9AY 153465097 IC50 > 100000 nM T05089 CZ9A4F 153465098 IC50 > 100000 nM T05089 C76TJD 155535190 IC50 > 100000 nM T44458 D05SBO 46220502 IC50 = 57 nM T44458 D00RYA 16750271 IC50 = 36 nM T44458 D00UZR 5330286 IC50 = 794.33 nM T44458 D05ADP 160355 IC50 = 230 nM T44458 D07DTV 11338033 IC50 = 10 nM T44458 D07KBM 124155204 IC50 < 4 nM T44458 D08HOM 46207586 IC50 > 10000 nM T44458 D0CY1B 6420138 Ki = 480 nM T44458 D0DX4J 67409219 IC50 < 100 nM T44458 D0LF1U 5287969 Ki = 3 nM T44458 D0P0KN 16739650 IC50 = 3 nM T44458 D0S5RC 3025986 Ki = 4 nM T44458 D0D3PX 46926350 IC50 = 4 nM T44458 CB9F1O 447961 Ki = 4 nM T44458 C6A3LY 447962 Ki = 575 nM T44458 C4GPF6 5329921 IC50 = 550 nM T44458 CVX20F 9842276 IC50 = 107 nM T44458 CVE1W8 10024433 Ki = 1153 nM T44458 C1KX3P 10248401 Ki > 10000 nM T44458 C9J3RM 10320107 Ki = 448 nM T44458 CMY9D2 10340715 Ki = 559 nM T44458 CC3L8Z 10430000 Ki = 2605 nM T44458 C4VX1Q 11065484 IC50 > 10000 nM T44458 C3F6UB 11300082 IC50 = 29 nM T44458 C3S2FX 11357740 IC50 = 31 nM T44458 CIWA03 11632150 Ki = 11 nM T44458 CEV5X2 11646645 Ki = 9 nM T44458 C2CVI7 11647020 Ki = 564 nM T44458 C93KHF 11718021 Ki = 6 nM T44458 CJSV21 11744184 Ki = 1472 nM T44458 COW2S0 13422576 IC50 = 300 nM T44458 C7BS2R 16037674 IC50 > 10000 nM T44458 CB2H4D 16037675 IC50 = 2500 nM T44458 C5VPH9 16129448 IC50 = 5330 nM T44458 C1BLP4 23582519 IC50 = 218 nM T44458 CO79TF 24809803 IC50 = 10 nM T44458 C4BV0K 25169528 IC50 = 770 nM T44458 CE65CO 25169529 IC50 = 120 nM T44458 CN8VA1 25190892 IC50 = 17 nM T44458 CIN53D 25190893 IC50 = 83 nM T44458 CL1Q0M 25190896 IC50 = 96 nM T44458 CX4Z1H 25195254 IC50 = 355 nM T44458 C5HZF2 44413509 IC50 = 2.5 nM T44458 C3D4FG 44413527 IC50 = 26 nM T44458 C3VRO9 44557921 IC50 > 10000 nM T44458 CSJ14N 44563119 IC50 = 1500 nM T44458 CXEW65 44563120 IC50 = 680 nM T44458 C5VQG1 44563155 IC50 = 810 nM T44458 CK4GU3 44563156 IC50 = 1600 nM T44458 CNS69D 44563157 IC50 = 370 nM T44458 CKU49O 44563158 IC50 = 270 nM T44458 CK8F3Q 44563194 IC50 = 3200 nM T44458 CH48EY 44563195 IC50 = 4100 nM T44458 C4W9HX 44580967 IC50 > 10000 nM T44458 CSE67T 44581007 IC50 > 10000 nM T44458 CB0F8O 44581008 IC50 = 3500 nM T44458 CKU1P7 44581009 IC50 > 10000 nM T44458 C2ZIH5 44581010 IC50 > 10000 nM T44458 C9HAU7 44581033 IC50 > 10000 nM T44458 CL6Y9J 44581034 IC50 > 10000 nM T44458 CGO1J5 46830766 Ki = 348 nM T44458 CF7HK2 46830767 Ki = 337 nM T44458 C2HJ1X 46830768 Ki = 264 nM T44458 C1SI2W 49830586 IC50 = 630.96 nM T44458 C06MKW 49839561 Ki = 111 nM T44458 CCL3R5 49867929 IC50 = 2180 nM T44458 C37NKO 67129970 IC50 > 10000 nM T44458 CK80LJ 67130050 IC50 > 10000 nM T44458 C9WY2P 67383875 Ki = 108 nM T44458 CYI75G 68678653 IC50 > 30000 nM T44458 C7GRV2 68755406 IC50 > 10000 nM T44458 C3GTU1 69762142 IC50 = 911 nM T44458 C65YEI 71618220 IC50 = 385 nM T44458 CF7R0Y 71682057 IC50 = 5300 nM T44458 CBE67N 71731769 IC50 = 7450 nM T44458 C7K5EN 73776233 IC50 = 1070 nM T44458 C7VA5U 78161839 IC50 = 1711 nM T44458 C2Y1RF 78162193 IC50 < 50 nM T44458 C4NM0V 78162195 IC50 < 50 nM T44458 CWR57U 78357763 IC50 = 134 nM T44458 CQ2SU8 78673832 IC50 > 30000 nM T44458 CE0W9R 78673833 IC50 > 30000 nM T44458 C8N7GL 87123415 IC50 = 1200 nM T44458 C3Q0LD 87767734 IC50 = 6 nM T44458 C26KEM 91262312 IC50 > 10000 nM T44458 CWE9I2 91664021 IC50 > 10000 nM T44458 CW58AE 91664022 IC50 = 2200 nM T44458 CB25UZ 91664023 IC50 = 1500 nM T44458 CX58DI 118716791 IC50 > 30000 nM T44458 CD9X2B 118716796 IC50 > 30000 nM T44458 C2YJ0O 118716797 IC50 > 30000 nM T44458 CL3UO9 118716798 IC50 > 30000 nM T44458 C71BAM 118716799 IC50 > 30000 nM T44458 CU4EL6 118716806 IC50 > 30000 nM T44458 CO83PN 122181013 IC50 = 15000 nM T44458 C69ULZ 122181014 IC50 = 160 nM T44458 CN14DV 122181015 IC50 = 120 nM T44458 CIG8Y1 122181016 IC50 > 10000 nM T44458 CRJS41 122181017 IC50 = 1000 nM T44458 CVB03H 122181018 IC50 = 1500 nM T44458 C6SJ3X 122181019 IC50 > 10000 nM T44458 C58CJI 122181022 IC50 > 10000 nM T44458 CG2Z8B 122181023 IC50 = 210 nM T44458 CC2G8N 122181024 IC50 = 3100 nM T44458 CM2DU7 122181025 IC50 > 10000 nM T44458 C5YB3O 122181096 IC50 = 350 nM T44458 CV5BQ9 122181097 IC50 = 2000 nM T44458 CO57LX 125501624 IC50 = 4 nM T44458 CSFJ98 126511854 IC50 = 270 nM T44458 COF75Z 126970673 IC50 = 450 nM T44458 C1SP3H 127030849 IC50 = 240 nM T44458 CC1VO7 127047444 IC50 > 25000 nM T44458 CDJQ32 127051599 IC50 = 37 nM T44458 C2LWZ1 129318964 IC50 = 1430 nM T44458 C46KZG 131704449 IC50 = 150 nM T44458 CCPZ70 131704452 IC50 = 6100 nM T44458 CJ3M5I 134137436 Ki = 17 nM T44458 C1MTG5 134543905 IC50 > 200 nM T44458 CQP51Y 134814484 EC50 < 100 nM T44458 CH29JY 135398514 IC50 = 350 nM T44458 C7PJ6X 135566704 IC50 > 30000 nM T44458 CH3M4B 137083628 IC50 > 30000 nM T44458 CJA07O 137083629 IC50 > 30000 nM T44458 C9F8PX 137083630 IC50 > 30000 nM T44458 C3DNL6 137349544 IC50 = 1100 nM T44458 CU9O3A 137628639 IC50 = 1.9 nM T44458 CI1E8V 137634241 IC50 > 10000 nM T44458 CGB8T4 137645179 IC50 = 20 nM T44458 CQ82UE 137662204 IC50 = 5000 nM T44458 CVU63L 139582016 IC50 = 370 nM T44458 C8PH9S 139582017 IC50 = 13000 nM T44458 CXS4L8 145975683 IC50 = 870 nM T44458 CB2J4N 145989210 IC50 = 4 nM T44458 C5YW8Q 145993622 IC50 = 10 nM T44458 CYHW79 155530843 IC50 = 20 nM T44458 C8OC5N 155537111 IC50 = 20 nM T44458 CETH36 155557337 IC50 > 200 nM T44458 CLXN40 155565350 IC50 = 26 nM T44458 D00ERW 44444843 Ki > 1644 nM T44458 D00HSJ 10275789 IC50 = 1.4 nM T44458 D03DZO 11715767 IC50 = 34 nM T44458 D0GN5Z 5281295 IC50 = 2160 nM T44458 D0J4ON 135473382 IC50 = 9 nM T44458 D0T8NU 16757525 IC50 = 28 nM T14912 D00PBX 49846579 Ki > 444 nM T14912 D02OZK 11404337 EC50 = 500 nM T14912 D06ETI 24978538 Ki < 1 nM T14912 D06XCP 131634760 Ki = 0.17 nM T14912 D0I5DP 118910268 Ki = 0.06 nM T14912 D0Q7AG 53240420 IC50 > 50000 nM T14912 D0Z0HH 3503 Ki = 162 nM T14912 D03TTE 135513044 Ki = 25 nM T14912 D0B1UL 136002683 Ki = 230 nM T14912 D0CR9A 136183441 Ki = 310 nM T14912 D0L8WH 11228183 Ki > 1 nM T14912 CI6DR8 4563 IC50 > 8.9 ug.mL-1 T14912 CK4N7S 6293 Ki = 1620 nM T14912 C45RGA 10331 Ki > 1000000 nM T14912 CQ6B2R 11768 Ki = 270 nM T14912 CS9PU3 27695 Ki = 160000 nM T14912 CVD64E 36941 Ki = 47800 nM T14912 CDZI90 67584 IC50 = 34000 nM T14912 CL89PK 72899 Ki > 1000000 nM T14912 CJUW83 95696 Ki = 103000 nM T14912 CF6GB0 96894 Ki = 2850 nM T14912 CK70FI 97423 Ki = 99000 nM T14912 CZF61E 124216 IC50 = 280000 nM T14912 C6FK9M 196978 Ki = 2270 nM T14912 CS5UA3 297061 Ki = 10410 nM T14912 C9Z5QR 307964 Ki = 131000 nM T14912 C0SMD7 339231 IC50 > 10 ug.mL-1 T14912 CCV98F 577543 Ki = 109000 nM T14912 CA10YW 597283 IC50 = 160000 nM T14912 CT42DP 620146 Ki = 81000 nM T14912 C3OG4Q 694880 Ki > 27000 nM T14912 C76CAZ 719016 Ki = 86000 nM T14912 CGH82E 739884 Ki = 59000 nM T14912 CMP56I 815185 Ki = 40000 nM T14912 C08YVK 819258 Ki = 22000 nM T14912 CYE67S 865778 Ki = 52000 nM T14912 C7GY1X 869152 Ki > 10000 nM T14912 CHY9D5 925045 IC50 > 25000 nM T14912 C07POK 992585 Ki = 3560 nM T14912 CK3ON2 992588 Ki = 1550 nM T14912 CLJ98I 992590 Ki = 810 nM T14912 C3S4QD 1068457 IC50 = 11000 nM T14912 CSK95Z 1068481 IC50 > 25000 nM T14912 CZC19M 1068514 IC50 = 21000 nM T14912 CQ4S3J 1068532 IC50 = 149 nM T14912 CKRU94 1076742 IC50 = 20000 nM T14912 C3OP8Z 1184112 Ki = 3130 nM T14912 CJ2KV9 1184138 Ki = 4230 nM T14912 C1AV5K 1184140 Ki = 730 nM T14912 C76DFX 1190498 IC50 = 7300 nM T14912 CMF16D 1309516 Ki = 820 nM T14912 C6U1DV 1315064 IC50 > 25000 nM T14912 CGAM30 1582605 Ki = 1550 nM T14912 CX21SU 1819997 Ki = 1060 nM T14912 CR4UC2 2058961 IC50 = 7170 nM T14912 C1V6BU 2227421 IC50 = 9000 nM T14912 C1G7KW 2324749 IC50 = 19000 nM T14912 C5EY8P 2763910 Ki = 8190 nM T14912 CC74TR 2771353 Ki = 3800 nM T14912 CGF4E6 2961169 IC50 > 25000 nM T14912 CMG0F6 2961623 IC50 = 400 nM T14912 C9G3PF 2966040 IC50 = 2400 nM T14912 CPS79F 3163284 Ki = 102000 nM T14912 CPJ5Y3 3701653 IC50 = 130000 nM T14912 C5A7UV 3850940 IC50 = 13000 nM T14912 C6DHN0 3855232 IC50 = 5500 nM T14912 C1NX4W 3969372 Ki = 12000 nM T14912 C06AJP 4192838 IC50 = 22000 nM T14912 CJ1E6P 4613756 IC50 = 73000 nM T14912 CMJ1G4 5018231 IC50 = 23000 nM T14912 CHP03C 5355594 Ki > 50000 nM T14912 C6KS5N 5356316 Ki > 50000 nM T14912 C85WLD 5927890 Ki > 50000 nM T14912 CIH5Q3 5955473 Ki = 21000 nM T14912 C3JX7W 6484626 Ki = 214000 nM T14912 CYFD93 6713806 Ki = 12000 nM T14912 CSM21W 6874071 Ki = 1000 nM T14912 CMTP73 7515143 Ki = 10000 nM T14912 CR8G5J 7566371 Ki = 7000 nM T14912 CI7MW0 9852185 IC50 = 790 nM T14912 CP5W2H 10019325 Ki > 50000 nM T14912 CZ8B7D 10348509 IC50 > 10 ug.mL-1 T14912 CV71EJ 10955342 IC50 = 190000 nM T14912 CV1X4J 11031986 Ki = 312 nM T14912 CDZ09C 11245319 Ki > 50000 nM T14912 CDAT72 11433190 Ki > 10000 nM T14912 C1FO6C 11500877 IC50 = 35 nM T14912 CV4JK3 11502754 IC50 > 100000 nM T14912 C8U6YE 11527635 IC50 = 39 nM T14912 CCU2Q9 11801671 IC50 > 10 ug.mL-1 T14912 C8TQX1 12158631 Ki = 398.11 nM T14912 CN9EL4 13044634 Ki = 23000 nM T14912 CP9GZ6 13548111 IC50 = 3300 nM T14912 CJMH83 14157895 Ki > 50000 nM T14912 CN0TX9 14716643 Ki = 131000 nM T14912 CQG83E 15101872 IC50 = 3300 nM T14912 C5X0CE 16380269 Ki > 50000 nM T14912 CW5KI7 16482412 Ki = 1130 nM T14912 CV7HC8 16645886 Ki = 136000 nM T14912 CZVP08 16735295 Ki = 18 nM T14912 CO38KM 16735541 Ki = 1690 nM T14912 CTMN68 17543415 IC50 = 18000 nM T14912 CJG10L 20099598 IC50 = 7200 nM T14912 C2I1RJ 20100040 IC50 = 2200 nM T14912 C4WTI8 21576164 IC50 > 10 ug.mL-1 T14912 CR2F6A 21637536 IC50 > 10 ug.mL-1 T14912 CHR5G0 22548322 IC50 = 1800 nM T14912 C49JYU 22683787 Ki = 60000 nM T14912 CJR38Q 22774194 IC50 = 12000 nM T14912 C7OZI2 24797083 Ki = 10.1 nM T14912 C5NI1B 24798804 IC50 > 1000 nM T14912 C9MNJ7 24800647 Ki = 4570.88 nM T14912 CNQF59 24800648 Ki = 380 nM T14912 CJB1U9 24801007 Ki = 338.84 nM T14912 CN61HR 24801008 Ki = 150 nM T14912 CP18YW 25058454 IC50 > 30000 nM T14912 CMS0Z5 25058455 IC50 > 100000 nM T14912 C7GHE9 25099966 Ki = 4400 nM T14912 CIX21K 25099968 Ki = 1700 nM T14912 C4Z7CN 25100119 Ki = 330 nM T14912 C2N5PJ 25100121 Ki = 2900 nM T14912 CS2WU4 25100442 Ki = 300 nM T14912 C74OSJ 25100590 Ki = 260 nM T14912 CHYW16 25144061 Ki = 9 nM T14912 CM56CP 25144613 Ki = 130 nM T14912 CQ2RZ7 25144887 Ki = 35 nM T14912 CZ57GE 25144888 Ki = 160 nM T14912 CHS0R4 25144889 Ki = 150 nM T14912 CZ12DX 25229694 Ki = 520 nM T14912 C7L9FT 25990016 Ki > 50000 nM T14912 CNU41H 40852065 Ki > 27000 nM T14912 CK78WE 42601456 Ki = 250 nM T14912 CY9CP3 42613557 Ki = 174 nM T14912 CA9JF3 44191246 IC50 = 3200 nM T14912 C2FXA3 44191638 IC50 = 1100 nM T14912 CXO2S9 44191694 IC50 = 300 nM T14912 CHT92S 44191696 IC50 = 590 nM T14912 C83UCJ 44191750 IC50 = 350 nM T14912 CMS39X 44191815 IC50 = 830 nM T14912 C0J3RT 44192144 IC50 = 230 nM T14912 C97RQU 44192145 IC50 = 780 nM T14912 C57VCY 44224066 IC50 = 330 nM T14912 CH2E4R 44609307 Ki = 370 nM T14912 CGTF35 45272228 IC50 > 10 ug.mL-1 T14912 C8FU1I 45273079 IC50 > 10 ug.mL-1 T14912 CG2NH7 46236925 IC50 = 200 nM T14912 C78NZA 46236926 IC50 = 240 nM T14912 C4FIO9 46831414 IC50 = 11400 nM T14912 C61KTO 46831415 IC50 = 12500 nM T14912 C9TIX2 49830849 Ki = 290 nM T14912 C6TAV4 51002999 Ki = 1281 nM T14912 C0J4PO 51003000 Ki = 122 nM T14912 CVBX71 51003001 Ki = 99 nM T14912 CJUQ29 51003002 Ki = 122 nM T14912 CMQ3U0 51003003 Ki = 967 nM T14912 CJ07CN 51003059 Ki = 1511 nM T14912 CE84DN 51003060 Ki = 842 nM T14912 CWQ69L 51003061 Ki = 151 nM T14912 CG57VY 51003062 Ki = 82 nM T14912 CHW3N9 51003063 Ki = 91 nM T14912 C9USE3 51003064 IC50 = 585 nM T14912 C8BZY6 51003123 IC50 = 5 nM T14912 CQ2X4R 51003124 Ki = 49 nM T14912 C2ZT6I 51354614 IC50 > 1000 nM T14912 C73DOP 51354615 IC50 > 1000 nM T14912 CNA1W2 51354616 IC50 > 1000 nM T14912 C4Q3YN 51354902 IC50 > 1000 nM T14912 CON3Q1 51354903 IC50 > 1000 nM T14912 C52OHD 51354904 IC50 > 1000 nM T14912 CM3CU0 51355193 IC50 > 1000 nM T14912 C3NI5T 53213045 Ki = 51000 nM T14912 CE23VN 53213046 Ki = 35000 nM T14912 CW9IN1 53234692 Ki = 4160 nM T14912 CWTA43 53234693 Ki = 3020 nM T14912 CTPX94 53234694 Ki = 3090 nM T14912 CC34HU 53234695 Ki = 2540 nM T14912 CHL4C7 53234842 Ki = 4100 nM T14912 CZ8TK7 53234845 Ki = 3110 nM T14912 CS1ZG8 53235008 Ki = 3270 nM T14912 C6BA1V 53235009 Ki = 1800 nM T14912 CV75RW 53235092 Ki = 3110 nM T14912 C2K5GP 53235093 Ki = 4030 nM T14912 C9JD1C 53235169 Ki = 7220 nM T14912 C3Q9IV 53473132 IC50 = 16630 nM T14912 CD7O1T 53473133 IC50 = 7260 nM T14912 C4EW9Y 53473224 IC50 = 2510 nM T14912 CI9Z3T 53473225 IC50 = 3560 nM T14912 CK96PJ 53473226 IC50 = 17790 nM T14912 CD0T9X 53473227 IC50 = 5080 nM T14912 CCP0W5 53473228 IC50 > 1000000 nM T14912 C98WGS 53473229 IC50 = 8370 nM T14912 C5T1HQ 53473314 IC50 = 7570 nM T14912 CP9JX1 53473315 IC50 = 8690 nM T14912 C9QA7I 53473316 IC50 = 5760 nM T14912 CS5CP0 53473317 IC50 = 3240 nM T14912 C5M2UV 53473318 IC50 = 7110 nM T14912 CSZ78K 53473319 IC50 = 9780 nM T14912 C4HF7T 53473387 IC50 = 3720 nM T14912 CNVH01 53473388 IC50 = 2480 nM T14912 CU3J2D 53473389 IC50 = 4760 nM T14912 CCH9R0 53473390 IC50 = 42590 nM T14912 CB2D9Z 53473391 IC50 = 13200 nM T14912 C78YZW 53473392 IC50 = 38810 nM T14912 C9Q0XS 53473478 IC50 = 4880 nM T14912 CX70AC 53473479 IC50 = 620 nM T14912 C6OTX3 53473480 IC50 = 6630 nM T14912 C1ME6Q 53473481 IC50 = 3180 nM T14912 CQHB31 53473482 IC50 = 3040 nM T14912 CHV0G1 53473570 IC50 = 3040 nM T14912 CN4O2V 53473571 IC50 = 3910 nM T14912 CSJ50X 53473572 IC50 = 140 nM T14912 C1O6KH 53473573 IC50 = 43220 nM T14912 C9L6JQ 53473574 IC50 = 25380 nM T14912 C9AYX8 53473660 IC50 > 1000000 nM T14912 C1GY0B 53473661 IC50 = 6300 nM T14912 C50AOR 53473662 IC50 = 220 nM T14912 C8KQ6V 54578933 Ki = 24 nM T14912 CRO6I8 54769781 Ki = 213 nM T14912 CZ1E8X 54769782 Ki = 445 nM T14912 C7WQI6 54769783 Ki = 149 nM T14912 CO7DE8 54769992 Ki = 375 nM T14912 CU4RQ6 56933429 IC50 > 2000 nM T14912 CNKE09 56933430 IC50 > 2000 nM T14912 CS3YP8 56933431 IC50 > 2000 nM T14912 C9CEO1 57338853 Ki = 1790 nM T14912 C38QHP 57339126 IC50 > 100000 nM T14912 C5XN9L 57394832 Ki = 3110 nM T14912 CSM8T4 57398377 Ki = 2290 nM T14912 CXP56B 57523339 IC50 > 10000 nM T14912 CX8EG1 57523340 IC50 > 10000 nM T14912 CC3KU7 57523369 IC50 > 10000 nM T14912 COA97D 57523370 IC50 > 10000 nM T14912 C61FYR 57523400 IC50 > 10000 nM T14912 CQ3L5W 57523401 IC50 > 10000 nM T14912 CH3I5T 57523430 IC50 > 100000 nM T14912 C8P2QI 57523431 IC50 > 100000 nM T14912 CX9BE7 57523432 IC50 > 10000 nM T14912 CF6IZ8 57523433 IC50 > 2000 nM T14912 C1YTI4 57523468 IC50 > 2000 nM T14912 C9AFI7 57523469 IC50 > 2000 nM T14912 C0OMZ9 57523470 IC50 > 2000 nM T14912 C4RDZ5 57523498 IC50 > 2000 nM T14912 CNFW46 59053624 IC50 > 10000 nM T14912 CBLR64 59447577 Ki > 440 nM T14912 C52IXR 60169703 IC50 > 100000 nM T14912 CN28ME 60169704 IC50 > 2000 nM T14912 CI13RU 60169705 IC50 > 10000 nM T14912 C49HLF 60169795 IC50 > 2000 nM T14912 CHAV90 60169796 IC50 > 2000 nM T14912 CI93MH 60171063 IC50 > 100000 nM T14912 C9VX1Y 61394197 IC50 > 25000 nM T14912 C8ZCV7 66575373 Ki = 0.45 nM T14912 CK8Q2I 67316207 Ki = 470 nM T14912 CDP69S 67442266 IC50 = 31000 nM T14912 C7ULB8 68863859 IC50 = 5000 nM T14912 CM3E4K 68938909 Ki = 1.8 nM T14912 C5M4OJ 68940388 Ki = 1.5 nM T14912 C8DY5U 68941543 IC50 = 383 nM T14912 C2W5BS 70680244 Ki = 55 nM T14912 CF5OC7 70680245 Ki = 320 nM T14912 CJ3YR9 70684416 IC50 > 10000 nM T14912 CTYS31 70686561 IC50 > 10000 nM T14912 C8C7FS 71451698 EC50 = 2100 nM T14912 CD1N9X 71452025 Ki = 38 nM T14912 CU59ZI 71452026 Ki = 107 nM T14912 CE03NH 71453306 IC50 > 10000 nM T14912 CW4J8S 71453826 Ki = 53 nM T14912 CJA8N4 71455243 EC50 = 7900 nM T14912 COH24E 71455246 EC50 = 11600 nM T14912 CVC5F8 71455247 EC50 = 2300 nM T14912 C3TL5D 71459209 Ki = 56 nM T14912 CS69ET 71459210 Ki = 13 nM T14912 CUG8N7 71462421 EC50 = 3500 nM T14912 C7N0LI 71545001 Ki = 12500 nM T14912 C4MKL2 71545163 Ki = 9600 nM T14912 CVF0O2 71545164 Ki = 370 nM T14912 C03ACL 71545165 Ki = 9500 nM T14912 CW1C6I 71545166 Ki = 14600 nM T14912 C4E1FO 71545167 Ki = 1000 nM T14912 C3PIM0 71545168 Ki = 35000 nM T14912 C82YDN 71545169 Ki = 15000 nM T14912 CZ6WO4 71545325 Ki = 8800 nM T14912 C9S4RJ 71545326 Ki = 1900 nM T14912 C9M6SH 71545327 Ki = 16000 nM T14912 CNK35Q 71545328 Ki = 9800 nM T14912 CB2E6L 71545329 Ki = 9900 nM T14912 CAW6K1 71545330 Ki = 380 nM T14912 CF67LD 71545331 Ki = 1100 nM T14912 CHPJ72 71545486 Ki = 300 nM T14912 C89YZF 71545487 Ki = 7700 nM T14912 C3N1CZ 71545488 Ki = 7600 nM T14912 CFY19U 71545489 Ki = 5200 nM T14912 CWQJ74 71545490 Ki = 6400 nM T14912 CMZ64C 71545491 Ki = 7500 nM T14912 CW9DU1 71545492 Ki = 480 nM T14912 C2L8VP 71545646 Ki = 62000 nM T14912 C68BAC 71545647 Ki = 14000 nM T14912 C2Q7CA 71545648 Ki = 810 nM T14912 CMW3S0 71545649 Ki = 160 nM T14912 CL1XT7 71545650 Ki = 700 nM T14912 CS92IM 71545651 Ki = 190 nM T14912 CC7I6A 71545824 Ki = 75 nM T14912 C5L1KM 71545825 Ki = 66 nM T14912 CGL67T 71545826 Ki = 180 nM T14912 CA0FZ2 71545827 Ki = 140 nM T14912 CBW68J 71545828 Ki = 290 nM T14912 C8X2IV 71545829 Ki = 1300 nM T14912 CFLE52 71545992 Ki = 1600 nM T14912 CS14HM 71545993 Ki = 250 nM T14912 C0HP4B 71545994 Ki = 120 nM T14912 C2JB5K 71545995 Ki = 750 nM T14912 C6OQK8 71545996 Ki = 720 nM T14912 CY63CR 71545997 Ki = 3000 nM T14912 CGL94Z 71545998 Ki = 2500 nM T14912 C2ZJI6 71546153 Ki = 1200 nM T14912 CE9T5S 71546154 Ki = 410 nM T14912 C8H9OE 71546155 Ki > 500000 nM T14912 CP3Y2O 71548702 Ki = 170 nM T14912 C9ZMN5 71548703 Ki > 27000 nM T14912 C4TU2L 71548705 Ki = 20000 nM T14912 C41KGN 71548852 Ki > 27000 nM T14912 CFUR95 71548853 Ki = 5080 nM T14912 CUTC42 71548854 Ki = 1710 nM T14912 CGQ87K 71548855 Ki > 27000 nM T14912 CACN32 71548856 Ki = 2180 nM T14912 CRA43U 71548999 Ki > 27000 nM T14912 CS02CG 71549001 Ki = 380 nM T14912 CRM47B 71549002 Ki = 40180 nM T14912 C3NE6X 71549004 Ki = 59350 nM T14912 C72SIQ 71549135 Ki = 12530 nM T14912 CV3MN5 71549136 Ki = 5230 nM T14912 C37AJW 71549412 Ki = 2030 nM T14912 C36HPA 71549413 Ki = 74920 nM T14912 C2PK4T 71549414 Ki = 4420 nM T14912 CYIR97 71550101 Ki = 2220 nM T14912 CO68SD 71550812 IC50 = 26840 nM T14912 CWMX49 71575178 Ki = 6320 nM T14912 C7KGD6 71575179 Ki = 12600 nM T14912 CE6P9G 71575180 Ki = 3290 nM T14912 CH89RV 71575181 Ki = 2520 nM T14912 CA8GM0 71575182 Ki = 7090 nM T14912 C1LYO4 71575286 Ki = 4830 nM T14912 C0IF6E 71575287 Ki = 5310 nM T14912 C9WC0G 71575292 Ki = 467.74 nM T14912 CX3RW8 71575293 Ki = 223.87 nM T14912 CMT91V 71575294 Ki = 53.7 nM T14912 CR1J5Q 71575403 Ki = 190.55 nM T14912 CN2F9Z 71716725 IC50 > 10000 nM T14912 CXWU63 71716750 Ki = 90000 nM T14912 CN86BR 71717322 IC50 > 10000 nM T14912 CO1XU7 71717940 Ki = 860 nM T14912 CJ7ZB2 71719772 Ki = 15280 nM T14912 C2M3KV 72724194 Ki = 320 nM T14912 C3J5NW 72724333 Ki = 180 nM T14912 CRM08G 72793103 IC50 = 540 nM T14912 C6C8FO 72793104 IC50 > 100000 nM T14912 CX86EJ 72793174 IC50 > 30000 nM T14912 CY23TP 72793175 IC50 = 3200 nM T14912 CS5R9Y 72793176 IC50 = 610 nM T14912 CB6E4W 72793245 IC50 = 88 nM T14912 CA1X8P 73167580 IC50 = 500 nM T14912 CX8D2P 73213475 Ki = 1200 nM T14912 CO8G6C 73213476 Ki = 1600 nM T14912 CQ17EJ 73213477 Ki = 1900 nM T14912 CO6E8W 73213478 Ki = 560 nM T14912 CDO87T 73213545 Ki = 630 nM T14912 C9G8FB 73213546 Ki = 580 nM T14912 C2GKN6 73213617 Ki = 2200 nM T14912 C07IDZ 73214403 Ki = 6400 nM T14912 C7P6IE 73214474 Ki = 3300 nM T14912 C16QYZ 73214475 Ki = 940 nM T14912 C3E1VM 73214476 Ki = 1200 nM T14912 C58DAI 73214477 Ki = 990 nM T14912 C90NSV 73214548 Ki = 530 nM T14912 CEV7T0 73214549 Ki = 2200 nM T14912 CZ1SQ0 73214550 Ki = 740 nM T14912 CXJ1F6 73214551 Ki = 3200 nM T14912 C0TAJ1 73334912 Ki = 155 nM T14912 CSJ24B 73346580 IC50 = 500 nM T14912 CZ7SP9 73347969 Ki = 1981 nM T14912 C4L1GZ 73347970 Ki = 2816 nM T14912 CGRZ30 73349519 Ki = 3240 nM T14912 CYF5H4 73349609 IC50 > 25000 nM T14912 CTU5K9 73349610 IC50 = 7500 nM T14912 CY7KD2 73351068 Ki = 1214 nM T14912 C7Q3SW 73351069 Ki = 123 nM T14912 C8PA5N 73352636 IC50 = 1200 nM T14912 CJ8MA1 73355661 IC50 = 310 nM T14912 C56WFQ 73357106 Ki = 609 nM T14912 CSC6D9 73386712 Ki = 14 nM T14912 C60OQK 76310973 IC50 = 200 nM T14912 CEA8O5 76310974 IC50 = 150 nM T14912 CC9JG6 76310975 IC50 = 60 nM T14912 CIW32J 76310976 IC50 = 4900 nM T14912 C56LIG 76310977 IC50 = 1800 nM T14912 CEX7O4 76310978 IC50 = 1200 nM T14912 C0BD1Z 76318179 IC50 = 30 nM T14912 C3WKT7 76318180 IC50 > 25000 nM T14912 C5G3ZI 76321884 IC50 = 45000 nM T14912 CJ6DR8 76321885 IC50 = 670 nM T14912 C73NKA 76325518 IC50 = 6200 nM T14912 CV07UH 76325519 IC50 = 1100 nM T14912 C2SKV3 76325520 IC50 = 1000 nM T14912 CI0V1A 76325521 IC50 = 400 nM T14912 COYQ08 76329056 IC50 = 22000 nM T14912 C14LSY 76329057 IC50 > 25000 nM T14912 C6QEU5 76332731 IC50 = 3400 nM T14912 CBJ7O5 76332732 IC50 = 80 nM T14912 CTY8R6 76332733 IC50 = 780 nM T14912 C12XPO 76332734 IC50 = 570 nM T14912 CWB51G 76332735 IC50 = 37000 nM T14912 C3ZLR4 76336347 IC50 = 300 nM T14912 C0UN6L 76336348 IC50 = 110 nM T14912 CKHP71 84622107 Ki = 90000 nM T14912 CR2TL5 85468775 Ki = 79 nM T14912 C3J7XU 85898121 Ki = 2950 nM T14912 CTZH71 86278051 IC50 = 4500 nM T14912 CHL56P 86730609 Ki = 86980 nM T14912 C3C7QO 86765310 Ki = 180 nM T14912 CI9EB4 89486940 IC50 > 100000 nM T14912 CVA4U6 89487009 Ki = 1540 nM T14912 C29DIO 89493598 Ki = 1010 nM T14912 C2NHG7 89493672 IC50 = 170 nM T14912 CF1J4N 89493712 Ki = 24200 nM T14912 CZN0P6 90080177 Ki = 656 nM T14912 C9M5EH 90080930 Ki = 322 nM T14912 CMX73V 90082750 Ki = 66 nM T14912 C7ZK5R 90082757 Ki = 1098 nM T14912 CQG0K9 90082811 Ki = 116 nM T14912 CP27DA 90082843 Ki = 1015 nM T14912 CKQ2S9 90082856 Ki = 298 nM T14912 CNL82Z 90082885 Ki = 430 nM T14912 C3NT4E 90082933 Ki = 251 nM T14912 CT46NE 90083001 Ki = 79 nM T14912 CNP13Q 90083030 Ki = 361 nM T14912 C46TXB 90083070 Ki = 20 nM T14912 CZ6U2J 90083185 Ki = 36 nM T14912 CT51MA 90083384 Ki = 335 nM T14912 CES21F 90083807 Ki = 55 nM T14912 CGFK15 90083809 Ki = 374 nM T14912 CIOP24 90083847 Ki = 139 nM T14912 CBR82C 90083861 Ki = 118 nM T14912 CH3VW8 90083897 Ki = 46 nM T14912 C89KSG 90083900 Ki = 278 nM T14912 C48FWQ 90083913 Ki = 90 nM T14912 CAU0G7 90083916 Ki = 193 nM T14912 CB5T7V 90084010 Ki = 87 nM T14912 CZN69S 90084083 Ki = 209 nM T14912 C7K2OY 90085536 Ki = 202 nM T14912 CK13AL 90085582 Ki < 10 nM T14912 C3T7BU 90085661 Ki = 231 nM T14912 COIA01 90085667 Ki = 209 nM T14912 CYLD27 90085696 Ki = 311 nM T14912 C9KR2C 90085736 Ki = 18 nM T14912 CI82NL 90085789 Ki = 119 nM T14912 C9IOB3 90085790 Ki = 432 nM T14912 CWAQ29 90085798 Ki = 655 nM T14912 CZQI28 90085826 Ki = 336 nM T14912 C04RXD 90316425 IC50 = 6100 nM T14912 C9J0CU 90342584 Ki = 2350 nM T14912 CV0AI7 90645495 Ki = 14000 nM T14912 CP06VM 90645496 Ki = 13000 nM T14912 CN24WU 90645497 Ki = 5200 nM T14912 CU8G4Y 90645498 Ki = 5900 nM T14912 C79THC 90656473 Ki = 550 nM T14912 C9YMU8 90656474 Ki = 240 nM T14912 C5I0PN 90656475 IC50 = 30200 nM T14912 CS31TR 90656476 Ki = 3790 nM T14912 C16KYS 90656477 Ki = 210 nM T14912 C12JEQ 91754241 Ki = 310 nM T14912 C5T9WD 94962278 Ki = 3620 nM T14912 CB0C4L 100690587 IC50 = 10000 nM T14912 CG24NQ 113098709 IC50 = 11000 nM T14912 CY3B0M 117275529 Ki = 18000 nM T14912 C4L9PU 118394580 Ki = 2.1 nM T14912 CD1QU8 118394588 Ki = 620 nM T14912 CP1X5K 118394589 Ki = 12 nM T14912 C2KQL1 118394601 Ki = 70 nM T14912 C9D1HV 118394606 Ki = 73 nM T14912 COYT16 118394615 Ki = 22 nM T14912 CBH3X1 118394618 Ki = 42 nM T14912 CUC1A4 118394619 Ki = 35 nM T14912 C4OTK1 118394623 Ki = 1.1 nM T14912 CHL0X1 118394626 Ki = 1.3 nM T14912 CAT47U 118394627 Ki = 1 nM T14912 CH8EQ9 118394659 Ki = 15 nM T14912 C05UPS 118394660 Ki = 9.6 nM T14912 CQ9DO1 118394677 Ki = 51 nM T14912 C5Z7XJ 118394681 Ki = 37 nM T14912 CGB9K5 118394682 Ki = 9.9 nM T14912 CI4T9N 118394685 Ki = 1.8 nM T14912 CNZ98G 118394699 Ki = 5.9 nM T14912 CY03IG 118394714 Ki = 23 nM T14912 CO40GK 118394721 Ki = 0.21 nM T14912 CIWY53 118394752 Ki = 47 nM T14912 C80KST 118394755 Ki = 570 nM T14912 CQ2I6F 118394756 Ki = 6.6 nM T14912 CFB9E0 118394766 Ki = 72 nM T14912 CJ6H4B 118394771 Ki = 17 nM T14912 CJ4WN5 118394779 Ki = 0.77 nM T14912 CXK64G 118394788 Ki < 7 nM T14912 C0GU4A 118394799 Ki = 11 nM T14912 CXB95M 118394806 Ki = 7.2 nM T14912 CKY8B2 118394807 Ki = 19 nM T14912 CJ58RP 118394818 Ki = 3.3 nM T14912 C4BI5A 118394823 Ki = 8.2 nM T14912 C80PUK 118394830 Ki = 9.6 nM T14912 C7HW0Y 118394836 Ki = 7.1 nM T14912 CE28ZO 118394843 Ki = 1.4 nM T14912 C91HQJ 118394848 Ki = 2.1 nM T14912 CQ15WJ 118394861 Ki = 12 nM T14912 CEF57G 118394864 Ki = 96 nM T14912 CZ39LF 118394865 Ki = 5.8 nM T14912 CC63UJ 118394876 Ki < 7 nM T14912 CT07OA 118394883 Ki = 12 nM T14912 CJ3B1P 118394895 Ki = 29 nM T14912 CIF46C 118394899 Ki = 24 nM T14912 C4K2JQ 118394913 Ki = 20 nM T14912 C53SNK 118394928 Ki = 48 nM T14912 C8UI9R 118394929 Ki = 31 nM T14912 C7KQT1 118394936 Ki = 69 nM T14912 C0T8GV 118394938 Ki = 22 nM T14912 C95GFD 118394942 Ki = 21 nM T14912 C3BQH4 118394951 Ki = 1.3 nM T14912 C85XVU 118394956 Ki = 7.6 nM T14912 CJH5O2 118394966 Ki = 27 nM T14912 CS2OR4 118394981 Ki = 8.7 nM T14912 CQ6Z8L 118406835 Ki = 1 nM T14912 CQT5W4 118406840 Ki = 0.77 nM T14912 CDX01Z 118406845 Ki = 2.4 nM T14912 C1P5AS 118406879 Ki = 4.9 nM T14912 CY1L9S 118406932 Ki = 0.31 nM T14912 CCI9J3 118406938 Ki = 43 nM T14912 CU47MW 118406940 Ki = 35 nM T14912 CBTM73 118406950 Ki = 1.8 nM T14912 CA7DW1 118406955 Ki = 0.7 nM T14912 CEOY82 118406960 Ki = 0.5 nM T14912 CW4K9Y 118406985 Ki < 1 nM T14912 C1O2ZX 118406988 Ki = 21 nM T14912 CPN23M 118406995 Ki = 0.65 nM T14912 C25TXW 118406996 Ki = 94 nM T14912 CEM24R 118406997 Ki = 1.2 nM T14912 CO1I7F 118407001 Ki = 130 nM T14912 CRX71A 118407022 Ki = 3200 nM T14912 C6LD2E 118407025 Ki = 2.9 nM T14912 CR80SJ 118407054 Ki = 1000 nM T14912 C2YF3O 118407086 Ki < 1 nM T14912 C0ZD3F 118521981 Ki = 53 nM T14912 C5XU9T 118522002 Ki = 148 nM T14912 C17ZUW 118522034 Ki = 91 nM T14912 CWE96A 118522037 Ki = 269 nM T14912 CHL0D3 118704913 Ki = 0.36 nM T14912 C8JGF6 118723013 Ki = 20000 nM T14912 CL1H0C 118723159 IC50 > 25000 nM T14912 C2TQ9L 118723160 IC50 > 50000 nM T14912 CFD7Z3 118723161 IC50 > 50000 nM T14912 C0XLN5 118723162 IC50 > 50000 nM T14912 CIS76T 118723163 IC50 > 50000 nM T14912 CVW41F 118723164 IC50 > 25000 nM T14912 C2JL8B 118723165 IC50 = 4100 nM T14912 CEL7Q0 118723166 IC50 = 21300 nM T14912 CBGY31 118723167 IC50 = 10000 nM T14912 CF17KU 118723168 IC50 > 50000 nM T14912 CEC7S8 118723169 IC50 > 50000 nM T14912 CSE54F 118728679 Ki = 86 nM T14912 C1QW4O 118728680 Ki = 66 nM T14912 C8XBN6 118728695 Ki = 63 nM T14912 C37NXV 118728696 Ki = 74 nM T14912 C9SLX5 118734954 Ki = 2.3 nM T14912 CR3U9V 118734955 Ki = 2 nM T14912 C1MFK7 118734956 Ki = 0.24 nM T14912 C5W2EA 118734957 Ki = 0.43 nM T14912 C4CP6R 118734958 Ki = 0.2 nM T14912 CA5Y7S 118734959 Ki = 0.31 nM T14912 CO8IZ0 118734960 Ki = 0.48 nM T14912 CW3Y1M 118737139 Ki = 18000 nM T14912 CU5S7Y 118737140 Ki = 3000 nM T14912 CO5K1H 118737141 Ki = 4000 nM T14912 C8HLR2 118737142 Ki = 1600 nM T14912 C40BQS 118737143 Ki = 120 nM T14912 C9BJR5 118737144 Ki = 110 nM T14912 C4G0TJ 118737145 Ki = 88 nM T14912 CNW6B0 118737146 Ki = 170 nM T14912 CLV10W 118737147 Ki = 74 nM T14912 CW29QH 118737148 Ki = 61 nM T14912 CRE89M 118737149 Ki = 150 nM T14912 C51KLE 118737150 Ki = 200 nM T14912 C0EA6G 118737151 Ki = 410 nM T14912 CPS8Z2 118737152 Ki = 210 nM T14912 CQ8M7Y 118737153 Ki = 71 nM T14912 C1ERH8 118737154 Ki = 110 nM T14912 C0NVR4 118737155 Ki = 65 nM T14912 CN7ZE6 118737156 Ki = 40 nM T14912 CP9MA5 118737157 Ki = 3 nM T14912 C2FOD3 118737158 Ki = 9 nM T14912 CEOC01 118737159 Ki = 0.454 nM T14912 CD6F7T 118910208 Ki = 0.05 nM T14912 C74NIY 118910215 Ki = 0.051 nM T14912 C42NRL 118910252 Ki = 0.14 nM T14912 C1H4DT 118910314 Ki = 0.04 nM T14912 C5XF0Y 121487966 IC50 = 237 nM T14912 CYN41X 121487972 IC50 = 162 nM T14912 C2N5KC 121487974 IC50 = 59.5 nM T14912 CTDA65 121487976 IC50 = 5.96 nM T14912 CYZ15O 121487977 IC50 = 4.7 nM T14912 CV0YR6 121487978 IC50 = 3.4 nM T14912 CZW49H 121487984 IC50 = 4.2 nM T14912 CUX2N7 122193137 Ki = 720 nM T14912 CDJE95 122193145 Ki = 700 nM T14912 C5S6PU 122193146 Ki = 1600 nM T14912 CA0KR9 122194475 Ki = 2900 nM T14912 C4ODZ9 122194476 Ki > 50000 nM T14912 CXTI31 122194478 Ki > 50000 nM T14912 CM7Y4S 122194479 Ki = 2300 nM T14912 CA45FG 122194480 Ki = 9300 nM T14912 C9SRV7 122194632 Ki = 3200 nM T14912 CUI60T 122194634 Ki = 3900 nM T14912 CNK8M7 122194635 Ki = 3700 nM T14912 C3Q7ND 122197581 Ki = 0.19 nM T14912 C76SBJ 122622651 Ki = 3400 nM T14912 CR19KU 122622656 Ki = 770 nM T14912 CFR02M 122622711 Ki = 87 nM T14912 CY2J6L 122622713 Ki = 1700 nM T14912 C0AYP2 122622799 Ki = 2600 nM T14912 CE4MG7 122622800 Ki = 1500 nM T14912 C0KP5W 122622803 Ki = 810 nM T14912 CIH4M1 122622824 Ki = 4700 nM T14912 CBFO10 122622827 Ki = 570 nM T14912 C6JOM4 122622922 Ki = 2000 nM T14912 CY9OL2 122623097 Ki = 220 nM T14912 C59MST 122623143 Ki = 90 nM T14912 C9YU0H 122623413 Ki = 840 nM T14912 CJ5P7N 122623425 Ki = 2700 nM T14912 C1R4UJ 122633925 Ki = 950 nM T14912 C26QUL 122633937 Ki = 13100 nM T14912 CX0N1V 126480720 Ki = 2500 nM T14912 C9QMC6 126480721 Ki = 34300 nM T14912 CM8SV0 126480722 Ki = 5030 nM T14912 CME8O4 126480723 Ki = 50300 nM T14912 CPV4H1 126480725 Ki = 23400 nM T14912 CM2OV0 126480726 Ki > 500000 nM T14912 CFS3X4 126480728 Ki = 31 nM T14912 C9TH3Q 126480729 Ki = 420 nM T14912 C2DF1E 126480732 Ki = 21000 nM T14912 CL4I2A 126480733 Ki = 120 nM T14912 C53RCO 126480736 Ki = 117 nM T14912 CY4HD9 126480737 Ki = 26900 nM T14912 CE4XG9 126480738 Ki = 3860 nM T14912 CI81TC 126480739 Ki = 8500 nM T14912 C71SZN 126480740 Ki = 1540 nM T14912 C20LKB 126480743 Ki = 2760 nM T14912 C9QJ0D 126480748 Ki = 566 nM T14912 CZF4Y9 126480749 Ki = 487 nM T14912 C0KI9X 126480779 Ki = 4540 nM T14912 CT5AP0 126480780 Ki = 11200 nM T14912 CJ25OH 126480781 Ki = 4580 nM T14912 CU58YJ 126480782 Ki = 1880 nM T14912 CX1D6L 126480784 Ki > 500000 nM T14912 CGDJ94 126480785 Ki = 6840 nM T14912 CHW0E3 126480786 Ki = 5640 nM T14912 CPN58B 126480787 Ki = 7310 nM T14912 CA1FE6 126480788 Ki = 284 nM T14912 C2FKU9 126480789 Ki = 3410 nM T14912 CMKN31 126480790 Ki = 106000 nM T14912 C6VK8A 126480791 Ki = 173 nM T14912 CX8EH4 126480820 Ki = 80 nM T14912 C6X1ID 126480821 Ki = 114 nM T14912 CUV13O 126480822 Ki = 335 nM T14912 CN6H1F 126480823 Ki = 79 nM T14912 CUL02S 126480864 Ki = 1910 nM T14912 CXF94P 126480867 Ki = 56300 nM T14912 C4KD8M 126480868 Ki = 33 nM T14912 CXK61D 126480870 Ki = 11900 nM T14912 CLCI06 126480871 Ki = 4050 nM T14912 C8IO2N 126480872 Ki = 22200 nM T14912 CDI79Q 126480873 Ki = 4490 nM T14912 C3VJ5L 126480874 Ki = 82 nM T14912 CSC41P 126480875 Ki = 1150 nM T14912 CH67EN 126480877 Ki = 54000 nM T14912 CY1Q2D 126480878 Ki = 25700 nM T14912 C3M2RF 127030077 Ki = 117 nM T14912 CW1U5M 127030374 Ki = 16 nM T14912 CS26VD 127030375 Ki = 10 nM T14912 CE48SO 127030379 Ki = 116 nM T14912 CW0JU5 127030388 Ki < 10 nM T14912 CN6L9W 127030695 Ki < 10 nM T14912 C0P7FG 127030987 Ki < 10 nM T14912 C03SVJ 127031331 Ki = 5.6 nM T14912 CHQY05 127031601 Ki = 2.4 nM T14912 C38FBK 127031602 Ki = 8.5 nM T14912 CIG1C9 127031603 Ki = 5.6 nM T14912 COW3X7 127031604 Ki = 1.2 nM T14912 C4K1WF 127031637 Ki = 19 nM T14912 CCU25Z 127031889 Ki = 2.5 nM T14912 C3UQ5T 127031890 Ki = 1 nM T14912 CQM29K 127031922 Ki = 100 nM T14912 CN1P6Y 127032748 Ki = 0.78 nM T14912 CW2DY9 127032749 Ki = 5 nM T14912 C5JI4W 127033064 Ki = 7 nM T14912 CER6M1 127033065 Ki = 10 nM T14912 CWY3K5 127033066 Ki = 2.9 nM T14912 CJZT46 127033067 Ki < 10 nM T14912 CJ2G6T 127033347 Ki < 10 nM T14912 CC6W5Z 127034471 Ki = 28 nM T14912 CN28OB 127034472 Ki = 782 nM T14912 CU3M7W 127034736 Ki = 8400 nM T14912 CQN8U5 127034737 Ki > 10000 nM T14912 CRU8S4 127034738 Ki > 10000 nM T14912 C95KTS 127034931 Ki > 10000 nM T14912 CUM3Q0 127035099 Ki > 10000 nM T14912 CYD17J 127035100 Ki > 10000 nM T14912 CGV45K 127035101 Ki > 10000 nM T14912 CEI73Z 127035102 Ki > 10000 nM T14912 C7MSI1 127035245 Ki > 10000 nM T14912 C8SHK4 127035480 Ki > 10000 nM T14912 C63PWT 127045713 Ki = 635 nM T14912 CU75LD 127045714 Ki = 404 nM T14912 CV4K2N 127045715 Ki = 81 nM T14912 C9TS4I 127045716 Ki = 393 nM T14912 CUT8S3 127045927 Ki = 161 nM T14912 CVEJ14 127046716 Ki = 722 nM T14912 C4F2JM 127046867 Ki > 10000 nM T14912 C8R2OD 127046868 Ki = 2600 nM T14912 CW7KI2 127046869 Ki = 4520 nM T14912 CZ8C3V 127047003 Ki = 8110 nM T14912 C4D6XB 127047004 Ki > 10000 nM T14912 CL68JY 127047005 Ki = 451 nM T14912 CX6WE4 127047006 Ki = 371 nM T14912 C9FMI6 127047007 Ki = 2390 nM T14912 C9TCV7 127047008 Ki = 226 nM T14912 C8ZX0Y 127048637 Ki > 50000 nM T14912 C37JKG 127048679 Ki > 50000 nM T14912 CYV35M 127048680 Ki > 50000 nM T14912 CJU4W5 127048681 Ki > 50000 nM T14912 CO87AZ 127048682 Ki > 50000 nM T14912 CH1GS3 127048965 Ki > 50000 nM T14912 CY8UL9 127049010 Ki > 50000 nM T14912 CHKJ87 127049283 Ki > 50000 nM T14912 C6TXC2 127049765 Ki = 180 nM T14912 CHQ07L 127049966 Ki = 3000 nM T14912 C8AE6C 127049967 Ki > 50000 nM T14912 CTA3Q5 127049968 Ki > 50000 nM T14912 CW38OQ 127049969 Ki > 50000 nM T14912 CB94FP 127050258 Ki = 7000 nM T14912 CDX32Q 127050259 Ki = 20000 nM T14912 CWA3Z4 127050260 Ki = 40000 nM T14912 C8FQI3 127050261 Ki > 50000 nM T14912 C80EFV 127050689 IC50 = 1400 nM T14912 C3N1EK 127051469 Ki = 2000 nM T14912 CI67FD 127052984 Ki = 28000 nM T14912 CHO7B1 134131757 Ki > 10000 nM T14912 C81IYU 134131766 Ki = 440 nM T14912 CXTI23 134131779 Ki = 8100 nM T14912 CZNS20 134131978 Ki = 410 nM T14912 CL56ET 134132368 Ki = 4000 nM T14912 C2CH6A 134133054 Ki = 220 nM T14912 CBZ96D 134133726 Ki = 1600 nM T14912 CIW4C3 134134074 Ki = 680 nM T14912 CFR14T 134134268 Ki = 320 nM T14912 CFZ72B 134134421 Ki = 500 nM T14912 CG2Q6C 134134900 Ki = 340 nM T14912 CJ7RT9 134135886 Ki = 5400 nM T14912 CA7BD0 134136566 Ki = 720 nM T14912 C1IVM2 134136602 Ki = 580 nM T14912 CDU1N4 134136951 Ki = 460 nM T14912 CMX0O4 134137098 Ki = 790 nM T14912 C0MAL5 134137174 Ki = 590 nM T14912 CY3X1V 134137192 Ki = 740 nM T14912 C1D4WS 134137526 Ki = 60 nM T14912 C91HZY 134139104 Ki = 14000 nM T14912 C9YDM6 134139400 Ki = 300 nM T14912 C15BUK 134139593 Ki = 4700 nM T14912 CM12BW 134139667 Ki = 430 nM T14912 C9ME1S 134140038 Ki = 290 nM T14912 CCA2Q3 134140830 Ki = 800 nM T14912 CW62KM 134141206 Ki > 10000 nM T14912 C3SN9F 134141542 Ki = 710 nM T14912 CM0X8W 134141608 Ki = 800 nM T14912 CC9HR2 134142084 Ki = 770 nM T14912 C3UL2F 134142985 Ki = 780 nM T14912 CH4U1M 134142993 Ki > 10000 nM T14912 CNE2A9 134143774 Ki = 500 nM T14912 CSFE39 134144182 Ki = 630 nM T14912 C1TSH9 134144208 Ki = 1300 nM T14912 C8ISK2 134144684 Ki = 480 nM T14912 CR6O8E 134144927 Ki = 500 nM T14912 C82ONI 134145686 Ki = 540 nM T14912 C7A8CM 134146167 Ki = 560 nM T14912 C0SLU6 134148123 Ki = 4000 nM T14912 CL57VN 134150368 Ki = 330 nM T14912 C1UHN8 134151998 Ki = 77 nM T14912 C2VC8J 134152063 Ki = 5600 nM T14912 C7ZH8I 134152922 Ki = 830 nM T14912 CW4EP2 134153984 Ki = 6900 nM T14912 CDUI74 134154308 Ki = 260 nM T14912 C9ATX6 134154502 Ki = 660 nM T14912 CQ24RE 134154949 Ki = 2700 nM T14912 CZ9Q5K 134155175 Ki = 1300 nM T14912 C61URW 134155768 Ki = 1700 nM T14912 CSCN35 134156097 Ki = 2000 nM T14912 C5THB4 134156624 Ki = 780 nM T14912 CFG1Z7 134157505 Ki = 8600 nM T14912 C7POE3 134157520 Ki = 900 nM T14912 CV0QH3 134157581 Ki = 590 nM T14912 C2INR6 134828256 Ki = 0.03 nM T14912 CL98UM 135340006 Ki = 1600 nM T14912 C41AEU 135397733 IC50 = 42 nM T14912 CY1SE5 135691163 IC50 = 4720 nM T14912 CAV6J3 135741996 Ki = 37 nM T14912 C9MFV2 136002682 Ki = 210 nM T14912 C6FY0E 136002684 Ki = 310 nM T14912 CU0YE2 136032534 Ki = 2070 nM T14912 CASH13 136032535 Ki = 3930 nM T14912 C9RD0X 136032611 Ki = 270 nM T14912 CH1J4T 136126562 Ki = 121 nM T14912 CC09EN 136183442 Ki = 1370 nM T14912 CYJD84 136183443 Ki = 450 nM T14912 CF8HV7 136183446 Ki = 25 nM T14912 C9TM5X 136190478 IC50 = 79 nM T14912 C1P6OX 136190479 IC50 = 15 nM T14912 C7QX1I 136190480 IC50 = 39 nM T14912 CM3W4P 136196528 Ki = 85 nM T14912 CLI5Y9 136217517 IC50 = 37 nM T14912 C6DTX1 136217518 IC50 = 37 nM T14912 CNY2V7 136217519 IC50 = 2500 nM T14912 CL1H4O 136217520 IC50 = 521 nM T14912 CY31SM 136217522 IC50 = 1100 nM T14912 CQ76AY 136217524 IC50 = 50 nM T14912 C1BOF5 136217525 IC50 = 30 nM T14912 CAB04U 136217526 IC50 = 10 nM T14912 CO86YC 136217527 IC50 = 150 nM T14912 C2GM7B 136217528 IC50 = 78 nM T14912 C6P5FM 136217530 IC50 = 141 nM T14912 CO40EL 136217531 IC50 = 75 nM T14912 C1EY2P 136229638 IC50 = 4800 nM T14912 C4SW3Y 136244512 Ki = 5981 nM T14912 CCG19P 136252244 IC50 = 42 nM T14912 C08TLG 136501290 Ki = 308 nM T14912 C73CEN 137243602 Ki = 247 nM T14912 CCDU12 137283305 Ki = 276 nM T14912 C3GOU1 137283377 Ki = 178 nM T14912 CPX64S 137289939 Ki = 139 nM T14912 C1TG3H 137290260 Ki = 94 nM T14912 CX07FI 137300716 Ki = 195 nM T14912 C9M8EW 137300717 Ki = 579 nM T14912 C5WI8H 137376079 Ki = 1.6 nM T14912 C28KCE 137631924 Ki = 570 nM T14912 CLP4D9 137631972 Ki = 0.089 nM T14912 CA6G9O 137632354 Ki > 30000 nM T14912 CQJ1P3 137633217 Ki = 1870 nM T14912 CF2NR4 137633615 Ki = 1.1 nM T14912 CS58WX 137633877 Ki = 12530 nM T14912 CFU98I 137634219 Ki = 600 nM T14912 C0MNE4 137634568 Ki = 140 nM T14912 CZ5G1N 137634735 Ki = 2380 nM T14912 CKF09I 137634986 Ki = 0.46 nM T14912 C26NRZ 137635896 Ki = 480 nM T14912 CZK3V7 137635900 Ki = 3370 nM T14912 C9DGP1 137637706 Ki > 30000 nM T14912 CD59HQ 137638062 Ki = 200 nM T14912 CJXA06 137638594 Ki > 30000 nM T14912 CYUH68 137639245 Ki = 250 nM T14912 C03QBO 137639274 Ki = 11610 nM T14912 C49LFT 137640943 Ki = 1190 nM T14912 CTX58M 137641044 Ki = 72 nM T14912 CGA35P 137641809 Ki = 0.24 nM T14912 CUPA80 137641828 Ki = 800 nM T14912 CLK5Q0 137642497 Ki = 4420 nM T14912 C37BPQ 137643293 Ki = 1630 nM T14912 CEH43O 137643523 Ki = 12870 nM T14912 CBY3S6 137644084 Ki = 490 nM T14912 CP47JW 137644266 Ki = 2100 nM T14912 C47XFD 137645331 Ki = 2680 nM T14912 CUI1C9 137645455 Ki > 30000 nM T14912 CC2ZE6 137645584 Ki = 2000 nM T14912 C20MST 137646146 Ki = 5380 nM T14912 C6ZIY9 137647191 Ki = 150 nM T14912 CRB6Q3 137647824 Ki = 960 nM T14912 C0J7UQ 137648092 Ki = 310 nM T14912 CBZK34 137650357 Ki = 3240 nM T14912 CBY54T 137650975 Ki = 10260 nM T14912 CMTL76 137652432 Ki = 9890 nM T14912 CE7KN1 137652918 Ki = 4130 nM T14912 CX9A0P 137654155 Ki = 2.4 nM T14912 C9ODE7 137654292 Ki = 890 nM T14912 C1QH5C 137655888 Ki > 30000 nM T14912 CX04FN 137656103 Ki = 740 nM T14912 CX87VH 137657686 Ki = 110 nM T14912 CU2CO7 137657986 Ki = 7780 nM T14912 CHYZ26 137658993 Ki = 200 nM T14912 CV8Q9S 137659015 Ki = 3000 nM T14912 CFPI02 137659018 Ki = 2570 nM T14912 CYA56C 137659271 Ki = 8190 nM T14912 CCR1T5 137659702 Ki = 1500 nM T14912 CAIP72 137659871 Ki = 1490 nM T14912 CV32NC 137660040 Ki = 22 nM T14912 CDQ5I7 137660190 Ki = 530 nM T14912 C0R5IX 137660420 Ki = 360 nM T14912 C1HXW0 137661513 Ki < 1 nM T14912 CP5U6T 137661597 Ki = 880 nM T14912 CNR17U 137661896 Ki = 950 nM T14912 CU70QV 138320064 IC50 = 40 nM T14912 CS2P8V 138320065 IC50 = 300 nM T14912 CVU5Y8 138393391 IC50 = 100 nM T14912 CA2Z3C 138454270 IC50 = 145 nM T14912 C5I8TQ 138756809 Ki = 22000 nM T14912 C8VST0 138756810 Ki = 2800 nM T14912 C0Y4VQ 138756811 Ki = 51 nM T14912 CJA5H2 138756812 Ki = 19 nM T14912 CWC9I8 138756813 Ki = 46 nM T14912 CPDC83 138756814 Ki = 2400 nM T14912 CKC68Y 139035047 IC50 = 11810 nM T14912 CP7X6U 139035048 IC50 = 780 nM T14912 C6RHG5 139476933 Ki = 0.1 nM T14912 C1G3HA 141721113 Ki = 0.42 nM T14912 CJ24FY 141721128 Ki = 0.081 nM T14912 CS5M3A 141721326 Ki = 0.33 nM T14912 CA40OL 141733224 Ki = 500 nM T14912 CV8LZ4 141733231 Ki = 450 nM T14912 CTR98A 141733249 Ki = 190 nM T14912 C2L5DS 145704704 Ki = 0.06 nM T14912 C6RJC4 145704705 Ki = 0.1 nM T14912 CJD6B0 145704706 Ki = 0.1 nM T14912 CRL4X3 145704707 Ki = 0.5 nM T14912 CH56LR 145704709 IC50 = 27 nM T14912 CI8J3D 145712375 IC50 = 4450 nM T14912 CMBT97 145712377 IC50 = 5950 nM T14912 CEV0C1 145953621 Ki = 2900 nM T14912 C3YPX4 145955393 Ki = 180 nM T14912 CCD35Z 145956354 Ki < 1 nM T14912 C7NH1G 145960303 Ki = 480 nM T14912 CR0WE4 145964234 Ki = 10200 nM T14912 C0L9RV 145964301 Ki = 419 nM T14912 COW54K 145964985 Ki = 8780 nM T14912 C7A3OW 145965232 Ki = 2780 nM T14912 C39KCH 145966546 Ki = 1190 nM T14912 C81GBE 145966945 Ki = 791 nM T14912 C04ZLA 145967530 Ki = 2340 nM T14912 CRX49Y 145967615 Ki = 4430 nM T14912 C6QFS7 145967616 Ki > 100000 nM T14912 C37LSX 145967655 Ki = 7330 nM T14912 CA64VN 145967660 Ki = 10300 nM T14912 CV3B0I 145967679 Ki = 13700 nM T14912 C5BWQ9 145967827 Ki = 40000 nM T14912 C4SYN0 145968061 Ki = 9240 nM T14912 CAN5F7 145968086 Ki = 7600 nM T14912 C3RM6C 145968116 Ki = 38200 nM T14912 CEN24G 145968358 Ki = 9770 nM T14912 C7HFG5 145968553 Ki = 8470 nM T14912 CCU89G 145968866 Ki = 6100 nM T14912 CS1E2B 145968967 Ki = 845 nM T14912 CG8U5Q 145969619 Ki > 100000 nM T14912 C5DXG2 145969951 Ki = 7440 nM T14912 CJM6E9 145970016 Ki = 19700 nM T14912 CLV9P0 145970350 Ki = 40000 nM T14912 CGQZ85 145970445 Ki = 100000 nM T14912 CYL2A5 145970652 Ki = 9220 nM T14912 CMN20R 145971153 Ki = 28800 nM T14912 CO9ZL6 145974129 Ki = 878 nM T14912 C56WVO 145974190 Ki = 12700 nM T14912 CWM4I3 145975764 Ki = 290 nM T14912 CM7G6U 145975792 Ki = 1940 nM T14912 C9XW0V 145976399 Ki = 2220 nM T14912 C12OSZ 145976540 Ki = 2130 nM T14912 CANX56 145977143 Ki = 1000 nM T14912 CXA76V 145977281 Ki > 100000 nM T14912 CG7I2O 145977960 Ki > 100000 nM T14912 C53OIY 145978226 Ki > 100000 nM T14912 C8J6QL 145978663 Ki > 100000 nM T14912 C6UVF9 145984310 Ki = 530 nM T14912 C5YH9I 145986580 Ki = 10900 nM T14912 CT8HL1 145989038 Ki = 40000 nM T14912 CCVP03 145994390 Ki = 94 nM T14912 C6PK1O 149610503 IC50 = 83 nM T14912 CUA74Q 153054039 Ki = 0.2 nM T14912 CJU6Q9 153341035 IC50 = 153 nM T14912 CX4F8J 153341235 Ki = 0.09 nM T14912 CCH6V2 153341378 Ki = 0.37 nM T14912 CH8QG4 155510354 Ki = 0.07 nM T14912 CVIW75 155511069 IC50 = 153 nM T14912 CL9HJ7 155511905 IC50 = 16010 nM T14912 CUX09D 155512545 Ki = 260 nM T14912 CIFA19 155512582 Ki = 0.11 nM T14912 CM8N5P 155513065 Ki = 0.1 nM T14912 C0S6NF 155513117 IC50 = 2800 nM T14912 CK25AN 155513849 Ki = 440 nM T14912 CBG8V7 155513976 Ki = 530 nM T14912 C9Z8FQ 155514893 Ki = 44000 nM T14912 CSE5N8 155515531 IC50 = 470 nM T14912 CTE3V7 155515598 Ki = 44000 nM T14912 CQ91VM 155515783 Ki = 300 nM T14912 CCZY53 155516133 Ki = 330 nM T14912 C8O3XM 155516217 IC50 = 1900 nM T14912 CJ7A1D 155516576 Ki = 27000 nM T14912 C8O3PF 155517190 IC50 = 10 nM T14912 C37INJ 155517782 IC50 = 7100 nM T14912 CP6J5F 155518107 Ki = 6000 nM T14912 C63PXN 155518333 IC50 = 690 nM T14912 CB37YD 155518816 IC50 > 10000 nM T14912 CB0C5P 155518916 IC50 = 10 nM T14912 CN28SY 155519167 IC50 = 4200 nM T14912 C6DOS2 155519264 Ki = 0.7 nM T14912 CLP32K 155519706 Ki = 59000 nM T14912 C91LSI 155520022 Ki = 24000 nM T14912 C2LT8A 155520283 Ki = 8100 nM T14912 CWO31S 155520968 Ki = 1990 nM T14912 CUJY40 155521076 Ki = 77000 nM T14912 CK7RM1 155521671 Ki = 220 nM T14912 C5G6CQ 155522270 Ki = 32 nM T14912 CR95IC 155522330 IC50 = 181 nM T14912 CE6QM8 155522510 Ki = 810 nM T14912 C1R8MS 155522698 Ki = 330 nM T14912 CKG0A6 155523132 Ki = 2000 nM T14912 C14OAS 155523253 Ki = 1 nM T14912 CZ8RY3 155523404 IC50 = 35 nM T14912 C5L4DX 155523696 Ki = 290 nM T14912 CQ6A8T 155524065 IC50 = 10640 nM T14912 C8V7CF 155524458 Ki = 490 nM T14912 C3HYI9 155524558 Ki = 7700 nM T14912 CN1U6Q 155524659 Ki = 61000 nM T14912 CQN1B8 155524663 Ki = 32800 nM T14912 C6W9LH 155524710 Ki = 53000 nM T14912 C9J0YL 155524932 IC50 = 7890 nM T14912 CWXZ56 155525506 Ki = 2.4 nM T14912 CLN6E5 155525940 IC50 = 8600 nM T14912 C01CQS 155526457 Ki = 110000 nM T14912 CXY0L3 155527670 Ki = 68000 nM T14912 CU2LZ8 155527825 Ki = 155 nM T14912 C02KFC 155527841 Ki = 1 nM T14912 CHA14B 155527900 Ki = 21000 nM T14912 CB89NA 155528220 Ki = 70400 nM T14912 C3AQO8 155529131 IC50 = 7000 nM T14912 CO0LH9 155529442 IC50 = 1500 nM T14912 CU9CX1 155529604 Ki = 200 nM T14912 CHI71P 155529809 IC50 = 153 nM T14912 CY6TH1 155530486 IC50 = 73 nM T14912 CRU28K 155530505 IC50 = 0.3 nM T14912 CF2KP7 155530563 Ki = 19000 nM T14912 CVE3A9 155530800 IC50 = 820 nM T14912 CD1WB3 155531298 Ki = 21 nM T14912 C95XMJ 155532216 Ki = 19000 nM T14912 CKT1X9 155534363 Ki = 0.28 nM T14912 C7L8AM 155534540 IC50 = 2030 nM T14912 C4ZNJ7 155534814 Ki = 27000 nM T14912 CHEO10 155535407 Ki = 48 nM T14912 CB3O4L 155535526 IC50 = 380 nM T14912 CV3L8Q 155536071 Ki = 8400 nM T14912 C5DSQ7 155536132 IC50 = 810 nM T14912 CNAR96 155536134 IC50 > 10000 nM T14912 CF6XB3 155536564 IC50 = 660 nM T14912 C7NRM6 155536808 Ki = 890 nM T14912 CK7UQ4 155537237 IC50 = 5960 nM T14912 C8HV9D 155537610 IC50 = 53 nM T14912 C0VBW2 155538516 IC50 = 15120 nM T14912 C39JKS 155538661 Ki = 15000 nM T14912 C7E4UB 155539057 IC50 = 420 nM T14912 CEAJ80 155539156 Ki = 51000 nM T14912 C6NI9J 155539696 Ki = 520 nM T14912 C5HAC4 155539927 Ki = 490 nM T14912 CW1EL8 155539938 Ki = 510 nM T14912 CEZ1F0 155540056 Ki = 58000 nM T14912 CC3A4H 155541877 Ki = 58 nM T14912 C81PLG 155542475 Ki = 45000 nM T14912 C8CEJ5 155542773 Ki = 50000 nM T14912 CUS28M 155542793 Ki = 73 nM T14912 CWHM15 155543101 IC50 = 210 nM T14912 CX5TO4 155543373 IC50 = 281 nM T14912 CJ4XS2 155543604 IC50 = 15 nM T14912 CI51ZW 155544348 IC50 = 920 nM T14912 CVBF96 155545115 Ki = 6100 nM T14912 CMI3D0 155545553 IC50 = 520000 nM T14912 C6TQ4X 155545656 IC50 > 8700 nM T14912 CL4HF7 155547093 Ki = 74 nM T14912 C4SM7J 155547389 IC50 = 7650 nM T14912 C0T4PZ 155547457 Ki = 110000 nM T14912 CD6IX3 155547704 Ki = 0.04 nM T14912 CPQ61U 155548293 IC50 = 112 nM T14912 C32SYB 155550004 Ki = 0.1 nM T14912 CAS76C 155551341 IC50 = 470 nM T14912 CO13SW 155552482 IC50 = 10 nM T14912 CS8N5R 155553044 IC50 = 1070 nM T14912 C7MTY0 155553176 IC50 > 25000 nM T14912 CH72LS 155553237 Ki = 480 nM T14912 CQAD72 155553397 IC50 = 17000 nM T14912 CKNH05 155553475 Ki = 0.1 nM T14912 C5YXT3 155553667 IC50 = 630 nM T14912 C5UX7I 155553713 Ki = 24000 nM T14912 C7E9FH 155554727 IC50 = 2.3 nM T14912 COE7Q1 155554903 IC50 = 300 nM T14912 CE2KQ4 155555867 IC50 = 3460 nM T14912 CGY43O 155556114 IC50 = 310 nM T14912 C4KGR1 155556368 Ki = 19000 nM T14912 C5U4EQ 155557291 IC50 = 1000 nM T14912 CNPA24 155558338 IC50 = 5400 nM T14912 CB2I1Z 155558410 IC50 = 7100 nM T14912 CUX0F2 155558443 IC50 > 10000 nM T14912 CHBE37 155560310 IC50 = 1510 nM T14912 CWRS76 155562189 Ki = 739 nM T14912 CC7BJ5 155562600 IC50 = 750 nM T14912 C6JC3K 155563087 Ki = 50000 nM T14912 CYIB91 155563107 Ki = 130000 nM T14912 CZW80Y 155563604 Ki = 76 nM T14912 CUY53S 155563898 IC50 = 1500 nM T14912 CG59ZN 155564461 IC50 = 9950 nM T14912 CEKN49 155565333 Ki = 0.05 nM T14912 CA68BM 155565390 IC50 = 2290 nM T14912 CF2A4I 155565463 Ki = 10000 nM T14912 C5Y0QF 155565915 IC50 = 9300 nM T14912 C79SGP 155566007 Ki = 100000 nM T14912 C3XP2F 155567783 Ki = 5210 nM T14912 C9KP8I 155568820 IC50 = 3500 nM T14912 C2W3PB 155568961 Ki = 0.05 nM T14912 C8CL3Z 155569283 IC50 > 10000 nM T14912 C21XOJ 155569465 IC50 = 149 nM T14912 CF8B9I 59053554 Ki = 4900 nM T14912 D00LHS 11455910 Ki = 260 nM T14912 D05RDP 992586 Ki = 180 nM T14912 D06VGD 6724 Ki = 57000 nM T14912 D0L6RV 3086109 IC50 = 2.4 ug.mL-1 T14912 D0V1DW 11952901 IC50 > 7.3 ug.mL-1 T14912 D0V7PX 454878 IC50 = 2600 nM T81547 CXCH42 124203831 IC50 = 501.19 nM T81547 C6LEZ9 127025652 IC50 > 25000 nM T81547 C2QN8R 127027156 IC50 = 800 nM T81547 CX6Z9U 127027780 IC50 = 1650 nM T81547 CWT17Q 127029348 IC50 = 410 nM T81547 CAL3O7 127029349 IC50 > 17000 nM T81547 CRHY95 127029612 IC50 = 316.23 nM T81547 CVR3Z1 127029613 IC50 > 18000 nM T81547 C14BIS 127029614 IC50 = 3162.28 nM T81547 C43GCS 127029619 IC50 = 190 nM T81547 CO1QL3 127029620 IC50 = 110 nM T81547 CUMN42 127029621 IC50 = 125.89 nM T81547 CAC06R 127029622 IC50 = 316.23 nM T84486 D08FJL 16681432 EC50 = 0.01 nM T84486 D0D8XY 5311010 Ki = 11 nM T84486 D0F4NS 119369 Ki = 660 nM T84486 D0M3FJ 439302 EC50 = 0.0046 nM T84486 D0N4OW 644077 EC50 = 0.1 nM T84486 D0U7SH 5311065 EC50 = 72 nM T84486 D04QZI 11340891 Ki = 0.63 nM T84486 D06VWL 10298385 Ki > 10000 nM T84486 D07EEN 172997 IC50 = 519 nM T84486 D09WYL 11634973 Ki = 0.1259 nM T84486 D0S3YN 53330936 EC50 = 2.399 nM T84486 D0SY9B 9895468 Ki = 1.514 nM T84486 D03RYS 5311500 Ki = 125 nM T84486 D08ORO 114904 Ki = 170 nM T84486 D08PAC 6918320 Ki = 4.6 nM T84486 D0A1KU 11683187 Ki = 9.5 nM T84486 D0Q8RX 9872389 Ki = 13 nM T84486 C0R7SI 449224 EC50 = 0.0091 nM T84486 CI82HM 999998 Ki = 470 nM T84486 C5F1ST 1103817 Ki = 14 nM T84486 CYHQ71 1103932 Ki = 90 nM T84486 CR4TP8 1107812 Ki = 620 nM T84486 CESI60 1134581 Ki = 100 nM T84486 C0WY8H 1134627 Ki = 800 nM T84486 CIAB57 1135733 Ki = 160 nM T84486 CZN48Y 1153909 Ki > 10000 nM T84486 C2HKQ3 1153925 Ki = 160 nM T84486 C1UAI6 1368921 Ki = 93 nM T84486 C0AB3Y 3601935 EC50 = 0.07943 nM T84486 C6C3XV 4017619 Ki = 50.12 nM T84486 C32BTU 4353841 Ki = 143 nM T84486 CQZF41 5002508 Ki = 199.53 nM T84486 C1C3LR 5014150 EC50 = 0.1 nM T84486 CQB93O 5306925 Ki < 10 nM T84486 C93WRU 9690136 Ki = 28 nM T84486 CO3SD6 9811830 EC50 > 10000 nM T84486 C4B6VD 9871105 IC50 = 68 nM T84486 COUA25 9938406 Ki = 1.4 nM T84486 CH2K5E 9954641 Ki > 10000 nM T84486 CIE8X5 9981665 Ki = 530 nM T84486 CG5AD1 10005688 Ki = 5.4 nM T84486 C5C3IS 10010253 Ki = 21 nM T84486 C8N7ET 10031014 Ki = 15.85 nM T84486 CIQT90 10054193 Ki = 25.12 nM T84486 CA07SF 10074886 Ki = 2 nM T84486 CK21XY 10078889 Ki = 5.1 nM T84486 CZPR64 10187625 EC50 = 640 nM T84486 CPEN43 10208363 Ki = 320 nM T84486 C3Q2JS 10259652 Ki = 4.5 nM T84486 C72BJX 10282736 EC50 = 2300 nM T84486 CRLZ04 10372918 Ki = 1.3 nM T84486 CTWG68 10411308 EC50 = 63 nM T84486 C1OIW6 10416272 Ki = 1.995 nM T84486 C0XHS9 10437668 Ki = 8 nM T84486 CR6VX2 10483105 Ki = 5.2 nM T84486 CJ8V4D 10507277 Ki = 11 nM T84486 CU4T8J 10507580 Ki = 13 nM T84486 CJ8C3T 10507800 Ki = 2.1 nM T84486 C4YB9E 10531717 Ki = 1.1 nM T84486 C9KDX3 10555563 Ki = 1 nM T84486 C42AVM 10556286 Ki = 1.2 nM T84486 C0L8KJ 10579644 Ki = 7 nM T84486 C0MBE3 10579886 Ki = 1 nM T84486 C2Z7RB 10587836 Ki < 10 nM T84486 CT50MD 10602875 Ki = 23 nM T84486 C4XF3E 10603831 Ki = 2.5 nM T84486 C7VS6M 10603858 Ki = 3.3 nM T84486 C58UPV 10627414 Ki = 5.1 nM T84486 C8NQ3K 10627984 Ki = 0.81 nM T84486 CWLZ69 10650710 Ki = 16 nM T84486 CP2C6H 10651225 Ki = 4.8 nM T84486 CK28TG 10651439 Ki = 4.2 nM T84486 C4PQ3B 10675476 Ki = 1.7 nM T84486 C41PCV 10675477 Ki = 2.3 nM T84486 CQ8J4S 10698572 Ki = 14 nM T84486 C9ML4W 10699322 Ki = 1.4 nM T84486 CSKL81 10699323 Ki = 6.7 nM T84486 CU7PT8 10721511 Ki = 29 nM T84486 CFH23E 10722297 Ki = 5.3 nM T84486 CDJH45 10722476 Ki = 2.5 nM T84486 C9B0GV 10723001 Ki = 0.82 nM T84486 C9X4ER 10746141 Ki = 5.6 nM T84486 C5HP1R 10746298 Ki = 2.3 nM T84486 CMP06T 10793202 Ki = 11 nM T84486 CE41AR 10817776 Ki = 1.5 nM T84486 C7KQE9 10837896 Ki = 82 nM T84486 CFZ3U0 10840517 Ki = 7.8 nM T84486 COU48N 10841081 Ki = 3.5 nM T84486 C0FJM7 11194023 Ki = 482 nM T84486 CO3A5Z 11240155 Ki = 1033 nM T84486 CC0KT1 11251777 Ki = 126 nM T84486 CUED54 11257380 Ki = 6 nM T84486 CY10OR 11260438 Ki = 1.995 nM T84486 C5OTG4 11274745 Ki = 664 nM T84486 C9T8BV 11286254 Ki = 223 nM T84486 CBH8C3 11295207 Ki = 0.631 nM T84486 CB6TF8 11297732 Ki = 164 nM T84486 CAY21S 11341369 Ki = 3.981 nM T84486 C70HTQ 11363194 Ki = 3.981 nM T84486 CYJ23D 11384094 Ki = 4 nM T84486 CWRG35 11385982 Ki = 79.43 nM T84486 CPND10 11389106 Ki = 206 nM T84486 CEM1X7 11400547 Ki = 1364 nM T84486 CMTX58 11408910 Ki = 5.012 nM T84486 C5VG6X 11421025 Ki = 0.1 nM T84486 CR4N5I 11465834 Ki = 0.07943 nM T84486 CM83DS 11468862 Ki = 1429 nM T84486 C37TNB 11475469 Ki = 14 nM T84486 C9SY7Q 11486351 Ki = 19 nM T84486 COC7Q9 11488952 Ki = 1 nM T84486 C4HJ6U 11495934 Ki = 12.59 nM T84486 CR5SH4 11502419 Ki = 2.2 nM T84486 C8M0VI 11511019 Ki = 1 nM T84486 C0HOR4 11519207 Ki = 1.585 nM T84486 CFA81S 11519251 Ki = 500 nM T84486 CPDL68 11525173 Ki = 316.23 nM T84486 C8K7EA 11534310 Ki = 158.49 nM T84486 C5PU0J 11538526 Ki = 4.2 nM T84486 C1SV4O 11547430 Ki = 0.05012 nM T84486 C4OUX7 11554957 Ki = 0.03162 nM T84486 CQ96XZ 11569194 Ki = 3.981 nM T84486 CCJ6K2 11569527 Ki = 0.631 nM T84486 C60DKW 11569672 Ki = 3.162 nM T84486 CY89CX 11570070 Ki = 0.03162 nM T84486 CI06OB 11570523 Ki = 3.981 nM T84486 CM15EB 11574636 Ki = 28.4 nM T84486 C4IH9D 11576272 Ki = 0.1 nM T84486 CL5B1V 11577215 Ki = 125.89 nM T84486 CFXV52 11577662 Ki = 5.012 nM T84486 CV1D0R 11577790 Ki = 25.12 nM T84486 CG7CL9 11578939 EC50 = 33 nM T84486 CP52SD 11590596 Ki = 0.5012 nM T84486 CT8KB7 11590614 Ki = 0.631 nM T84486 C4E8XS 11591519 Ki = 39.81 nM T84486 CCHO18 11598556 Ki = 63.1 nM T84486 C4TO5Q 11598736 Ki = 0.1259 nM T84486 C5UE4X 11605341 Ki = 0.03981 nM T84486 CNGW43 11606502 Ki = 158.49 nM T84486 CHB1N0 11612607 Ki = 3.981 nM T84486 C8NM7K 11613469 Ki = 6.31 nM T84486 CU9F1K 11618185 Ki = 2.6 nM T84486 CP0U2Q 11619807 Ki = 2750 nM T84486 CGF8K2 11619939 Ki = 100 nM T84486 CD2NZ0 11620428 Ki = 770 nM T84486 CFPR21 11625088 Ki = 5.4 nM T84486 C8D5PW 11626867 Ki > 10000 nM T84486 CA51GE 11627894 Ki = 79.43 nM T84486 CVEP03 11634960 Ki = 3.981 nM T84486 CXC7R1 11641200 Ki = 50.12 nM T84486 C60ODW 11641980 Ki > 10000 nM T84486 CN2D8B 11649100 Ki = 2.512 nM T84486 CB21DH 11656342 Ki = 25.12 nM T84486 CG4I7L 11662784 Ki = 0.3981 nM T84486 CBK9F2 11663715 Ki = 5.012 nM T84486 CQ4SX5 11667812 Ki = 17.5 nM T84486 CTMH91 11669836 Ki = 0.0631 nM T84486 COK9B6 11677260 Ki = 3.981 nM T84486 CY0HE4 11677610 IC50 > 100000 nM T84486 C97SUY 11677875 Ki = 2.512 nM T84486 C73DUI 11685100 Ki = 1.259 nM T84486 CPUR43 11685194 Ki = 1.995 nM T84486 C7AXL4 11691416 Ki = 50.12 nM T84486 C4OP8T 11691437 Ki = 0.05012 nM T84486 CT41LU 11692335 Ki = 510 nM T84486 C29LWS 11705315 Ki = 0.3981 nM T84486 CY54WJ 11706166 Ki = 158.49 nM T84486 CL4VK0 11719871 Ki = 0.07943 nM T84486 CIC93G 11740743 Ki = 30 nM T84486 C94OYW 11756466 Ki = 7.34 nM T84486 C4FL3O 11757835 Ki = 15.85 nM T84486 CFHQ73 11758421 Ki = 3.162 nM T84486 C91CIO 11815584 Ki = 25.6 nM T84486 CCQ01Y 11848692 Ki = 1 nM T84486 C8GC2P 11854507 IC50 > 100000 nM T84486 C4CTD2 14257660 EC50 = 70.79 nM T84486 CP46ID 15548578 Ki = 2.8 nM T84486 CC27MR 15548579 Ki = 4 nM T84486 C6TQ2F 15840423 Ki = 1 nM T84486 CMB5T2 15840433 Ki = 4.5 nM T84486 CTEW91 15951937 Ki = 7524 nM T84486 CHU5E4 16051933 Ki = 5 nM T84486 C7T2WZ 16062053 Ki = 350 nM T84486 C2Q9SA 18700090 Ki = 2.4 nM T84486 CFGI36 18700180 Ki = 0.86 nM T84486 C96PMU 18700187 Ki = 1.4 nM T84486 C4ZV6B 19690978 Ki = 1800 nM T84486 CQ73LX 19691006 Ki = 73 nM T84486 CJ3VW9 19691009 Ki = 54 nM T84486 CO45EK 21476314 Ki = 17 nM T84486 C6YU9B 21886866 Ki = 1.995 nM T84486 CG7JW4 22162609 EC50 = 0.12 nM T84486 COC73W 25212177 Ki = 0.7943 nM T84486 CJB78T 25212178 Ki = 12.59 nM T84486 CCX14Y 26434734 Ki > 1000 nM T84486 CY67HA 42611262 Ki = 0.7943 nM T84486 CM2D3L 44186995 Ki = 5.9 nM T84486 C78SLY 44214438 Ki = 2 nM T84486 CEX40M 44215484 Ki = 304 nM T84486 CB82ZC 44232512 EC50 = 0.04 nM T84486 CBV47F 44243143 Ki = 56 nM T84486 CDI2Q4 44247566 IC50 > 50118.72 nM T84486 C1ST4W 44274620 Ki = 794.33 nM T84486 CCQ4W9 44274621 Ki = 501.19 nM T84486 CR96PO 44274659 Ki = 39.81 nM T84486 CTSH82 44274660 Ki = 25.12 nM T84486 C87LZE 44274675 Ki = 100 nM T84486 CKUY40 44274724 Ki = 100 nM T84486 CR7S3D 44274883 Ki > 3162.28 nM T84486 CU7EQ6 44274915 Ki > 5011.87 nM T84486 CPV1O0 44274918 Ki > 5011.87 nM T84486 C3SYF2 44274927 Ki = 199.53 nM T84486 CRQ59U 44274928 Ki = 794.33 nM T84486 C08JOD 44274944 Ki = 79.43 nM T84486 CT9Z4B 44274970 Ki = 1584.89 nM T84486 C1VP5H 44274994 Ki = 100 nM T84486 C7UZL5 44275001 Ki = 794.33 nM T84486 CS2X4Z 44275002 Ki = 199.53 nM T84486 C7LTE5 44275003 Ki = 31.62 nM T84486 CAQZ90 44275012 Ki = 794.33 nM T84486 CI3B4T 44275026 Ki = 100 nM T84486 CWSZ16 44275048 Ki = 316.23 nM T84486 C8OQ2I 44275099 Ki = 19.95 nM T84486 CVI6Q3 44275104 Ki = 2.7 nM T84486 CAF32P 44275210 Ki = 390 nM T84486 CXT2P7 44275233 Ki = 9.8 nM T84486 C7GVH9 44275244 Ki = 240 nM T84486 CW7JM3 44275447 Ki = 1.1 nM T84486 C85JSQ 44275617 Ki = 33 nM T84486 C1CJ2V 44275618 Ki = 87 nM T84486 CRSA75 44278929 Ki = 199.53 nM T84486 C4OG9P 44278943 Ki = 19.95 nM T84486 C9BYG0 44278944 Ki = 199.53 nM T84486 CVC9E7 44278973 Ki = 794.33 nM T84486 CU9OY5 44278983 Ki = 125.89 nM T84486 CNTB12 44278986 Ki = 251.19 nM T84486 CPB8A7 44279000 Ki = 158.49 nM T84486 CX0E8C 44279151 Ki = 63.1 nM T84486 CH0P4D 44279165 Ki = 63.1 nM T84486 CIC2E1 44279168 Ki = 79.43 nM T84486 CKO01E 44279179 Ki = 6.31 nM T84486 C50FRI 44279238 Ki = 25.12 nM T84486 CTKC84 44279260 Ki = 794.33 nM T84486 CTMR53 44279329 Ki = 125.89 nM T84486 CRVE47 44279330 Ki = 125.89 nM T84486 CLNK46 44279348 Ki = 398.11 nM T84486 CA8T0B 44279368 Ki = 25.12 nM T84486 C20JXH 44279369 Ki = 3.981 nM T84486 CA0C8D 44279390 Ki = 15.85 nM T84486 CZ03MF 44279410 Ki = 3.162 nM T84486 CL41XB 44279411 Ki = 6.31 nM T84486 CL2VH6 44279433 Ki = 158.49 nM T84486 CM6UZ0 44279454 Ki = 398.11 nM T84486 C8NL6I 44279459 Ki = 25.12 nM T84486 CAP93K 44279482 Ki = 79.43 nM T84486 CM6V0D 44279483 Ki = 63.1 nM T84486 C7DSH6 44279485 Ki = 199.53 nM T84486 C9EQ0N 44279509 Ki = 316.23 nM T84486 CTM46I 44279519 Ki = 398.11 nM T84486 CBG89P 44279520 Ki = 0.5012 nM T84486 C03LWS 44279521 Ki = 7.943 nM T84486 CR4P7O 44279536 Ki = 25.12 nM T84486 CE9FP8 44279542 Ki = 3.162 nM T84486 CPZW45 44279555 Ki = 39.81 nM T84486 CA90KC 44279556 Ki = 794.33 nM T84486 C5WEK3 44279568 Ki = 63.1 nM T84486 CLI5J6 44279572 Ki = 1 nM T84486 CGM92O 44279573 Ki = 10 nM T84486 C9MJT4 44279574 Ki = 79.43 nM T84486 CO9JE1 44279580 Ki = 125.89 nM T84486 C08RBM 44279590 Ki = 3.981 nM T84486 CT89QV 44279607 Ki = 1.259 nM T84486 C9ABK0 44279637 Ki = 10 nM T84486 C9YSG3 44279676 Ki = 25.12 nM T84486 CZNW83 44279688 Ki = 100 nM T84486 CSP65I 44279689 Ki = 25.12 nM T84486 CF6HZ2 44279692 Ki = 15.85 nM T84486 C1DXH6 44279709 Ki = 7.943 nM T84486 CUH90A 44279710 Ki = 6.31 nM T84486 CVAY78 44279711 Ki = 6.31 nM T84486 C2QH3F 44279714 Ki = 794.33 nM T84486 CY78OA 44279752 Ki = 398.11 nM T84486 C0JRT4 44279772 Ki = 158.49 nM T84486 C3SJ2I 44279774 Ki = 199.53 nM T84486 CO6BS0 44279794 Ki = 794.33 nM T84486 CRB5X6 44279795 Ki = 63.1 nM T84486 CG24JT 44279846 Ki = 10 nM T84486 CO92JY 44279908 Ki = 1.995 nM T84486 C0ZD3O 44279909 Ki = 6.31 nM T84486 CH70NB 44279910 Ki = 2.512 nM T84486 CR3PO8 44279980 Ki = 50.12 nM T84486 C5P4NK 44279997 Ki = 100 nM T84486 CS38IL 44280013 Ki = 39.81 nM T84486 CH9C6W 44280354 Ki = 10 nM T84486 CE37MC 44280355 Ki < 3162.28 nM T84486 C1L6CB 44280356 Ki = 25.12 nM T84486 C3BS0D 44308876 Ki = 10 nM T84486 C2J8GK 44316235 Ki = 48.7 nM T84486 CIE6Y1 44316236 Ki = 556 nM T84486 C24NQS 44316241 Ki = 211 nM T84486 C52CNE 44334970 Ki = 17 nM T84486 CIS67O 44334971 Ki = 58 nM T84486 CSPU93 44334980 Ki = 160 nM T84486 CG1BN9 44334990 Ki = 73 nM T84486 CXH9Q7 44335148 Ki = 260 nM T84486 CK2H7V 44335184 Ki = 3.9 nM T84486 CU29TH 44335268 Ki = 15 nM T84486 C82YAS 44335300 Ki = 7.9 nM T84486 CTR03A 44356082 IC50 = 130 nM T84486 CNL9F6 44361387 Ki = 150 nM T84486 C5VCQ0 44361403 Ki = 200 nM T84486 C38FBJ 44361406 Ki = 130 nM T84486 CT0ZY3 44361521 Ki = 2100 nM T84486 CMG0N3 44361522 Ki = 24 nM T84486 C9E5JO 44393911 EC50 = 470 nM T84486 CDK52W 44393912 EC50 = 480 nM T84486 CZ4UB9 44393941 EC50 = 1500 nM T84486 C9JBI3 44393965 EC50 = 2800 nM T84486 CGW9Z6 44393998 EC50 > 10000 nM T84486 CUS19Z 44394044 EC50 = 430 nM T84486 C05DOG 44394045 EC50 = 2200 nM T84486 CZ4B0C 44394063 EC50 = 810 nM T84486 C81TIW 44404012 Ki = 10 nM T84486 CJF6U0 44404013 Ki = 31.62 nM T84486 CV92UP 44404027 Ki = 100 nM T84486 C89GPL 44404031 Ki = 158.49 nM T84486 CJUT58 44413575 Ki = 1.585 nM T84486 CS9B5A 44429266 IC50 = 51700 nM T84486 CS8M2O 44433363 IC50 = 1000 nM T84486 CLBA10 44433367 IC50 = 1000 nM T84486 CCI04H 44433372 IC50 = 1000 nM T84486 C9BDH6 44433375 IC50 = 1000 nM T84486 C8JLT7 44455964 Ki = 0.7943 nM T84486 CI14BY 44456003 Ki = 39.81 nM T84486 C78ISY 44456004 Ki = 1.259 nM T84486 CA8GN6 44456034 Ki = 6.31 nM T84486 CBA58Q 44456036 Ki = 6.31 nM T84486 CNGI92 44456070 Ki = 1.585 nM T84486 CHO6Q7 44456072 Ki = 12.59 nM T84486 CU1R3D 44456109 Ki = 1.259 nM T84486 CMJ25N 44456151 Ki = 0.1585 nM T84486 CDR9Y7 44456194 Ki = 0.7943 nM T84486 CQ27WK 44456229 Ki = 1.259 nM T84486 CO6N8J 44456270 Ki = 3.162 nM T84486 C1XE3I 44456352 Ki = 0.3981 nM T84486 CN2U1P 44456382 Ki = 6.31 nM T84486 C89DSK 44456383 Ki = 1 nM T84486 CPR06N 44456424 Ki = 1.995 nM T84486 CT62QR 44456469 Ki = 2.512 nM T84486 CO8NM3 44458614 IC50 = 130 nM T84486 C9SEC5 44459838 IC50 = 5 nM T84486 CEFB84 44459839 IC50 = 1 nM T84486 CLE7W0 44466239 IC50 > 19952.62 nM T84486 CKA3S0 44467347 IC50 > 50118.72 nM T84486 CPI04M 44563579 Ki > 10000 nM T84486 CVE5Y7 44571386 Ki = 15.85 nM T84486 CKE3V1 44571387 Ki = 63.1 nM T84486 C27LNY 44571388 Ki = 630.96 nM T84486 C5P0CU 44571389 Ki = 1000 nM T84486 CV0L4G 44571429 Ki = 79.43 nM T84486 CLI1M9 44571488 Ki = 1000 nM T84486 CL9SO6 44571489 Ki = 3162.28 nM T84486 C0SIU3 44571490 Ki = 6309.57 nM T84486 CC0A4K 44571491 Ki = 3.162 nM T84486 CXI7K6 44571492 Ki = 199.53 nM T84486 CU1XN0 44571529 Ki = 316.23 nM T84486 C4LIE5 44571530 Ki = 6309.57 nM T84486 C2QG0S 44572003 Ki = 3.162 nM T84486 CFD78Y 44572045 Ki = 63.1 nM T84486 CVH6I2 44572046 Ki = 630.96 nM T84486 C68RXE 44572047 Ki = 1995.26 nM T84486 C4ZET5 44572048 Ki = 125.89 nM T84486 C2U6JY 44572103 Ki = 7.943 nM T84486 CI8U6L 44572104 Ki = 79.43 nM T84486 CH0Z1M 44572105 Ki = 3162.28 nM T84486 CK1Z9I 44572106 Ki > 3162.28 nM T84486 C6D2RB 44572107 Ki = 39.81 nM T84486 CQ3V6N 44577873 Ki = 3 nM T84486 C2UQT0 44577874 Ki = 50 nM T84486 CMG70R 44577936 Ki = 56 nM T84486 CZD7E3 44577937 Ki = 16 nM T84486 C0HXR2 44577938 Ki = 43 nM T84486 COP3Q0 44577939 Ki = 17 nM T84486 C10ZLO 44577981 Ki = 84 nM T84486 C2WE1A 44577982 Ki = 2 nM T84486 CED75W 44577983 Ki = 232 nM T84486 C1E6GX 44577984 Ki = 537 nM T84486 C6R0AW 44578010 Ki = 201 nM T84486 CLCK14 44579399 Ki = 28 nM T84486 C6OK3X 44579400 Ki = 143 nM T84486 C0IHE7 44579401 Ki = 102 nM T84486 CU31MF 44579402 Ki = 190 nM T84486 CXOJ34 44579441 Ki = 144 nM T84486 CMW6Q7 44579442 Ki = 45 nM T84486 CM7HN8 44581240 Ki = 6.31 nM T84486 CG68XT 44581241 Ki = 3.162 nM T84486 CC5AT2 44581242 Ki = 1.995 nM T84486 C4FZQ9 44581266 Ki = 6.31 nM T84486 C0HF7U 44581267 Ki = 1.585 nM T84486 CO8YC5 44581268 Ki = 2.512 nM T84486 CB53IT 44581269 Ki = 3.981 nM T84486 CCM80P 44581647 Ki = 39.81 nM T84486 CNFH69 44581682 Ki = 39.81 nM T84486 CG36MZ 44581683 Ki = 63.1 nM T84486 CT1C8R 44581684 Ki = 63.1 nM T84486 C5NMB0 44581685 Ki = 125.89 nM T84486 CAJL21 44581686 Ki = 6.31 nM T84486 CW2CF8 44581687 Ki = 10 nM T84486 C1FH8I 44581718 Ki = 12.59 nM T84486 CKQO31 44581719 Ki = 12.59 nM T84486 C5GAR4 44581720 Ki = 12.59 nM T84486 CSZ70I 45103785 Ki = 2500 nM T84486 CK4XM7 45103786 Ki > 5000 nM T84486 CD7LT5 45268188 Ki = 198 nM T84486 C43IPM 45268191 Ki = 8.8 nM T84486 C0QDY7 45269934 Ki = 52.3 nM T84486 C23DQH 45270760 Ki = 253 nM T84486 CE06PJ 45271574 Ki = 12.5 nM T84486 CKS3B4 45271580 Ki = 14.6 nM T84486 C6XIZ7 45272485 Ki = 23.6 nM T84486 CHJ15D 45272491 Ki = 37.5 nM T84486 CCE9Z3 45273367 Ki = 9.4 nM T84486 CYQ36K 45483204 Ki = 316.23 nM T84486 C6LX7B 46225023 Ki = 114 nM T84486 C48JOB 46225048 Ki = 0.4 nM T84486 CX2S6L 46225049 Ki = 170 nM T84486 C70FCZ 46225050 Ki = 35.9 nM T84486 CIM9Y4 46225051 Ki = 31.8 nM T84486 CZ36XD 46225079 Ki = 28.5 nM T84486 CA6DS1 46225080 Ki = 17.9 nM T84486 COT65W 46225081 Ki = 5.8 nM T84486 C53ZIX 46225082 Ki = 207 nM T84486 CFLW87 46225083 Ki = 304 nM T84486 C7A8DU 46225116 Ki = 55.1 nM T84486 C4E8NX 46225117 Ki = 32.5 nM T84486 C3W6VI 46225118 Ki = 40 nM T84486 CT8LO5 46225153 Ki = 18.4 nM T84486 C98EDC 46233065 Ki = 844 nM T84486 CKET01 46233066 Ki = 245 nM T84486 C4K7AV 46830094 Ki = 11 nM T84486 CH4F6K 46830095 Ki = 14 nM T84486 CNU72P 46830096 Ki = 25 nM T84486 CS6JV3 46844643 Ki = 13.9 nM T84486 CDY4A0 46844644 Ki = 43 nM T84486 C3XYK5 46881859 Ki = 159 nM T84486 CZRH74 46881860 Ki = 237 nM T84486 CKR89V 46881861 Ki = 112 nM T84486 CF56RZ 46881862 Ki = 67.2 nM T84486 CA1WR6 46881890 Ki = 36.7 nM T84486 CNVS02 46881891 Ki = 48.4 nM T84486 CXV24Z 46881892 Ki = 41.4 nM T84486 CI3WD5 46881932 Ki = 19.7 nM T84486 C9Z0RU 46883829 Ki = 41 nM T84486 CP9IK8 46883830 Ki = 85 nM T84486 CSYZ34 46883831 Ki = 98 nM T84486 C3J8DL 46883832 Ki = 91 nM T84486 CSVJ29 46883884 Ki = 232 nM T84486 CPN1W9 46883885 Ki = 85 nM T84486 C2MK5O 46883886 Ki = 251 nM T84486 C8H5VB 46883887 Ki = 48 nM T84486 C4OYM9 46883888 Ki = 97 nM T84486 C2C5YZ 46883925 Ki = 84 nM T84486 CS35GM 46884413 Ki = 90 nM T84486 C0EMW2 46884414 Ki = 92 nM T84486 C3FUB6 46884437 Ki = 129 nM T84486 CM0RI1 46884438 Ki = 150 nM T84486 C4DP6I 46884439 Ki = 115 nM T84486 CB3X0J 46884440 Ki = 218 nM T84486 CXTE54 46884441 Ki = 620 nM T84486 C27WFG 46884478 Ki = 393 nM T84486 C3U2WD 46884479 Ki = 433 nM T84486 CB8WK2 46884480 Ki = 29 nM T84486 CUWG39 46934434 IC50 > 100000 nM T84486 CI9J7N 47177173 Ki = 396 nM T84486 CO9JL6 47177176 Ki < 10 nM T84486 CO4WH0 50941635 Ki = 5011.87 nM T84486 CMPE57 52941704 Ki > 10000 nM T84486 C5NMR0 52946086 Ki = 260 nM T84486 C6U3YN 52947354 Ki = 95 nM T84486 CHX2F3 52947410 Ki = 50 nM T84486 CBDS48 52949017 Ki = 5525 nM T84486 CM7V8G 53316559 Ki = 0.29 nM T84486 C0KBC6 53316694 Ki = 2511.89 nM T84486 CQ43EC 53316695 Ki = 25118.86 nM T84486 CN3X1M 53317550 Ki = 0.72 nM T84486 CH47QY 53317994 Ki = 3981.07 nM T84486 CEUQ37 53319051 Ki = 7.6 nM T84486 C8RSB7 53319199 Ki > 100000 nM T84486 C0E3DJ 53320505 Ki = 11.8 nM T84486 CO7BA3 53321697 Ki > 100000 nM T84486 CDJE61 53321821 Ki = 1404 nM T84486 C82IPZ 53321822 Ki > 100000 nM T84486 CS0Q9A 53323297 Ki = 6309.57 nM T84486 CLK0X6 53323298 Ki = 6309.57 nM T84486 CVB45I 53324622 Ki = 50118.72 nM T84486 C24KRL 53325929 Ki = 19952.62 nM T84486 C4TEY2 53358902 Ki > 10000 nM T84486 C5FA7N 53358903 Ki = 320 nM T84486 C63IVJ 53362154 EC50 > 10000 nM T84486 C21HMW 53362155 EC50 > 10000 nM T84486 CF60LM 53362156 EC50 > 10000 nM T84486 CGMY47 53362202 EC50 > 10000 nM T84486 C9V8RI 53362203 EC50 > 10000 nM T84486 CAL1Y3 53362204 EC50 > 10000 nM T84486 C6N5EX 53362257 EC50 > 10000 nM T84486 CS40QD 53362258 EC50 > 10000 nM T84486 CFWL28 53362259 EC50 > 10000 nM T84486 CNDR76 53362310 EC50 > 10000 nM T84486 COUH09 53362311 EC50 > 10000 nM T84486 C1MU4B 53362312 EC50 > 10000 nM T84486 CLRT87 53362368 EC50 > 10000 nM T84486 CG8J6H 53362369 EC50 > 10000 nM T84486 CD1N3U 53362370 EC50 > 10000 nM T84486 CRY95P 53362428 EC50 > 10000 nM T84486 C3TFA8 53362429 EC50 = 15.49 nM T84486 C4U1PT 53362430 EC50 = 32 nM T84486 C09KLV 53362488 EC50 = 31.62 nM T84486 CRX54F 53362489 EC50 = 43.65 nM T84486 C3KCI9 53362490 EC50 > 10000 nM T84486 CW32MV 53362546 EC50 > 10000 nM T84486 C5EG6T 53362547 EC50 > 10000 nM T84486 CUD9F0 53362548 EC50 > 10000 nM T84486 CVJ9U2 53362603 EC50 = 104.71 nM T84486 CMY7V4 53362604 EC50 > 10000 nM T84486 CK9V1G 53362605 EC50 > 10000 nM T84486 CCRZ83 53362670 EC50 > 10000 nM T84486 CYK9B3 53362671 EC50 = 257.04 nM T84486 CCK0P6 53362672 EC50 > 10000 nM T84486 CYG85M 53362729 EC50 = 9.1 nM T84486 C1IBT7 53362730 EC50 = 970 nM T84486 CI0F3Y 53362731 EC50 = 776.25 nM T84486 C3XW1F 53362732 EC50 > 10000 nM T84486 CYTJ92 53362793 EC50 > 10000 nM T84486 CQ9CD8 53362794 EC50 > 10000 nM T84486 CAN2C1 53362795 EC50 > 10000 nM T84486 CO4UA0 53362796 EC50 = 109.65 nM T84486 C0NSZ5 53362797 EC50 > 10000 nM T84486 CFJO73 53362798 EC50 = 860 nM T84486 C2RSW6 53362849 EC50 = 1200 nM T84486 C5K9YV 53362850 EC50 = 29 nM T84486 CB3AR7 53362851 EC50 = 29.51 nM T84486 C42SJF 53362852 EC50 > 10000 nM T84486 C8U6LX 53362853 EC50 > 10000 nM T84486 CH93SM 53362854 EC50 > 10000 nM T84486 C7RYJ0 53362909 EC50 = 104.71 nM T84486 CKV9D6 53362910 EC50 > 10000 nM T84486 CX9YM6 53362911 EC50 > 10000 nM T84486 C76TQB 53362913 EC50 > 10000 nM T84486 C5XCD8 53362914 EC50 > 10000 nM T84486 C8N0TX 53362915 EC50 > 10000 nM T84486 CU9X3P 53362962 EC50 > 10000 nM T84486 C61CNE 53362963 EC50 > 10000 nM T84486 CF30CI 53362964 EC50 > 10000 nM T84486 C6SB7W 53362965 EC50 > 10000 nM T84486 C32FZM 53362966 EC50 > 10000 nM T84486 CJ06TA 53362967 EC50 > 10000 nM T84486 C6AN7Y 53363015 EC50 = 180 nM T84486 C52IOF 53363016 EC50 = 173.78 nM T84486 C1SHU3 53363017 EC50 > 10000 nM T84486 CNA2L1 53364234 Ki = 380.19 nM T84486 C3L7RP 54580516 Ki = 20 nM T84486 CX1H3Z 54580518 Ki = 89 nM T84486 C7X4LI 54581307 Ki = 12.6 nM T84486 CB5R2M 54581528 Ki = 62 nM T84486 CR7GD2 54581529 Ki = 29 nM T84486 CUW8C7 54581530 Ki = 17 nM T84486 CD21EL 54581533 Ki = 115 nM T84486 C0ZNY9 54582318 Ki = 210 nM T84486 CQ7Z8U 54582526 Ki = 135 nM T84486 C7MP0S 54584254 Ki >= 10000 nM T84486 C73IGF 54584265 Ki = 29 nM T84486 CX5T1G 54584266 Ki = 21 nM T84486 CIGN05 54584267 Ki = 22 nM T84486 CC49GD 54584268 Ki = 3742 nM T84486 C9N2QH 54584476 Ki = 42 nM T84486 CD1A0H 54584477 Ki = 271 nM T84486 CXPY04 54584478 Ki = 28 nM T84486 CHR91Z 54585227 Ki = 179 nM T84486 C8YD0H 54585429 Ki = 45 nM T84486 C5N7VS 54585431 Ki = 170 nM T84486 C3MLH7 54586172 Ki >= 10000 nM T84486 C1N7LU 54586391 Ki = 45 nM T84486 C60DIQ 54586392 Ki = 7 nM T84486 CJ76VF 56657866 Ki = 0.4 nM T84486 C3T2HR 56657867 Ki = 0.34 nM T84486 CQG9J6 56657868 Ki = 0.17 nM T84486 C31CRV 56658409 EC50 > 10000 nM T84486 C6T3VC 56658416 EC50 = 3.3 nM T84486 C4FV1M 56664766 Ki = 9.4 nM T84486 CJ5FQ4 56664848 Ki = 0.29 nM T84486 C5V3ME 56664849 Ki = 0.25 nM T84486 C3SYC9 56665377 EC50 > 10000 nM T84486 CQN0G9 56668257 Ki = 6.24 nM T84486 CL07IK 56671720 Ki = 0.18 nM T84486 CU9DK4 56671721 Ki = 126 nM T84486 CSL0C7 56671723 Ki = 0.32 nM T84486 CNO51C 56675150 Ki = 0.09 nM T84486 C8GLI4 56675151 Ki = 1.8 nM T84486 C05JPT 56678446 Ki = 0.21 nM T84486 CNZU65 56682530 Ki = 102 nM T84486 C7JF1N 56949757 Ki = 0.3981 nM T84486 C8EMI5 56949758 Ki = 0.2512 nM T84486 CLKD45 56949759 Ki = 3.162 nM T84486 CQ8ZU3 56949760 Ki = 0.2512 nM T84486 C3VGA0 56949905 Ki = 1.585 nM T84486 CIU9N7 56949906 Ki = 0.3981 nM T84486 CUD7G6 56949907 Ki = 0.5012 nM T84486 CES5G4 56949908 Ki = 5.012 nM T84486 CH5I4O 56949909 Ki = 5.012 nM T84486 C87YDV 56950039 Ki = 0.3162 nM T84486 CM6VJ9 56950040 Ki = 0.0631 nM T84486 CF57NK 56950041 Ki = 0.07943 nM T84486 CODB85 56950042 Ki = 1 nM T84486 CLV0A3 56950043 Ki = 0.5012 nM T84486 C01VIN 56950167 Ki = 0.1585 nM T84486 CC2S8E 56950168 Ki = 1 nM T84486 C63UVA 56950169 Ki = 1.259 nM T84486 C3MTC5 56950170 Ki = 0.7943 nM T84486 CHRY19 56950171 Ki = 0.7943 nM T84486 CY47MH 56950311 Ki = 0.1995 nM T84486 CRAN69 56950449 Ki = 3.981 nM T84486 CY2JU8 56950450 Ki = 7.943 nM T84486 CLCK60 56950451 Ki = 15.85 nM T84486 C3BU6Q 56950452 Ki = 31.62 nM T84486 CUH08C 56950588 Ki = 0.02512 nM T84486 C2ORG7 56950589 Ki = 31.62 nM T84486 CXT5C1 56950590 Ki = 39.81 nM T84486 C21GOS 56950591 Ki = 39.81 nM T84486 CHG37B 57519947 Ki = 5.7 nM T84486 C0DB5C 57519948 Ki = 16 nM T84486 C15NPY 57520031 Ki = 28 nM T84486 C57LFR 57722466 Ki = 0.05012 nM T84486 CBTU57 67839485 Ki = 10.4 nM T84486 CD1IQ4 70685417 Ki = 10 nM T84486 CCTZ13 70685423 Ki = 78 nM T84486 C5TEF0 70694330 Ki = 158.49 nM T84486 CUD97X 71451749 Ki = 665 nM T84486 C7BCA6 71451750 Ki = 307 nM T84486 CJGO63 71451752 Ki = 495 nM T84486 C7T0WZ 71452693 Ki = 1000 nM T84486 C8KO3M 71453576 Ki > 10000 nM T84486 CG03VC 71455302 Ki = 808 nM T84486 C0IZ5N 71457081 Ki = 184 nM T84486 C1Q6RX 71462479 Ki > 10000 nM T84486 C4ZX0N 73345500 IC50 = 19000 nM T84486 CM8RF1 73346892 Ki = 856 nM T84486 CTVJ75 73346893 Ki = 1.5 nM T84486 CQW78U 73346990 Ki = 18 nM T84486 CY7IS2 73346991 Ki = 2.3 nM T84486 C2Y4UX 73348432 Ki = 91 nM T84486 C2FH9M 73349974 IC50 = 160 nM T84486 C7GDP3 73350017 Ki = 131 nM T84486 C8GQK9 73350823 Ki = 15 nM T84486 CQ8UO2 73351518 Ki = 224 nM T84486 CY4IW8 73351519 Ki = 143 nM T84486 CI7UV0 73353078 IC50 = 36000 nM T84486 CEB1I3 73354449 IC50 = 8 nM T84486 CG8AD1 73354500 Ki = 369 nM T84486 CLMY01 76073634 EC50 = 0.025 nM T84486 C53VYU 76685194 EC50 = 0.1 nM T84486 CLF3W5 90285421 EC50 = 0.07943 nM T84486 CNH3I0 90285477 EC50 = 520 nM T84486 C4VET9 90285722 EC50 = 47 nM T84486 C6MOJ3 90285806 EC50 = 753 nM T84486 CI76EP 90285817 EC50 = 2460 nM T84486 CZ6PL4 90285984 EC50 = 19 nM T84486 CTD92B 90286007 EC50 = 17 nM T84486 C59OHY 90286664 EC50 = 1570 nM T84486 CGZ9F1 90469608 EC50 > 10000 nM T84486 CRO49T 90469675 EC50 > 10000 nM T84486 CSKZ30 90469676 EC50 > 10000 nM T84486 CUL5F3 90663155 Ki = 0.6 nM T84486 CH8EA2 90663156 Ki = 0.3 nM T84486 CL45OR 90672737 EC50 = 13 nM T84486 CI2H0D 90679377 EC50 = 0.0067 nM T84486 C8U3HO 90680084 EC50 = 0.07 nM T84486 C45XGB 90680085 EC50 = 0.013 nM T84486 C2TGY7 118476332 EC50 > 10000 nM T84486 C76ONJ 118476338 EC50 = 230 nM T84486 C2RE7I 118476348 EC50 = 140 nM T84486 C5Z9SC 118476360 EC50 > 10000 nM T84486 C50MTE 118705579 Ki = 30 nM T84486 C9HX7Z 118705580 Ki = 963 nM T84486 CD0MS2 118716666 EC50 = 1570 nM T84486 CR3TZ0 118719818 EC50 = 0.05 nM T84486 CFG2V7 118719819 EC50 = 0.01 nM T84486 C4J6ZO 118719820 EC50 = 0.06 nM T84486 C9B2WS 118719821 EC50 = 0.01 nM T84486 CAFX95 118719822 EC50 = 0.98 nM T84486 CH74ZW 118719823 EC50 = 0.82 nM T84486 C7QI5K 118719824 EC50 = 0.06 nM T84486 CAP85S 118719825 EC50 = 0.21 nM T84486 CDR70N 118719826 EC50 = 0.37 nM T84486 CH0WU8 118719827 EC50 = 0.13 nM T84486 C1OMZ4 118719828 EC50 = 0.01 nM T84486 C72LOG 118719829 EC50 = 0.01 nM T84486 CD0P3Q 118719830 EC50 = 1.3 nM T84486 CAKC58 118719831 EC50 = 0.03 nM T84486 CIK48G 118719832 EC50 = 0.39 nM T84486 CDSK02 118719833 EC50 = 0.11 nM T84486 C9GSF2 118719834 EC50 = 0.12 nM T84486 CS89AW 118719835 EC50 = 0.01 nM T84486 CTWG46 118719836 EC50 = 0.15 nM T84486 COQ71F 118719837 EC50 = 0.01 nM T84486 CT3LR1 118719838 EC50 = 0.06 nM T84486 CX3R0J 118719839 EC50 = 1.3 nM T84486 CT3O7P 118719840 EC50 = 1.3 nM T84486 CW2F8P 118719841 EC50 = 0.46 nM T84486 CC9ZH4 118719842 EC50 = 0.12 nM T84486 C0LIH8 118719843 EC50 = 0.12 nM T84486 CYWM79 118719844 EC50 = 0.02 nM T84486 CGJ05D 118719845 EC50 = 0.0073 nM T84486 CH3DE8 118720259 EC50 = 0.11 nM T84486 C3DLZ2 118720260 EC50 = 0.02 nM T84486 COD37S 118720261 EC50 = 0.07 nM T84486 CPNB13 118720262 EC50 = 19 nM T84486 CW4Q3B 118720263 EC50 = 10 nM T84486 CI1SA4 118720264 EC50 = 0.11 nM T84486 CX2K6O 118720265 EC50 = 0.16 nM T84486 COHG04 118720266 EC50 = 0.96 nM T84486 CL2WY9 118720267 EC50 = 0.85 nM T84486 C53KXO 118720268 EC50 = 0.01 nM T84486 CH2T3S 118720269 EC50 = 0.13 nM T84486 C7KCE4 118720270 EC50 = 0.86 nM T84486 CEK5A6 118720271 EC50 = 0.12 nM T84486 C4OSR7 118720272 EC50 = 0.14 nM T84486 C2Z8IG 118720273 EC50 = 0.23 nM T84486 C3SD1R 118720274 EC50 = 0.09 nM T84486 CXGF75 118720275 EC50 = 0.11 nM T84486 CZ96MR 118720276 EC50 = 0.25 nM T84486 CM1V0E 118720277 EC50 = 0.07 nM T84486 CJB1T7 118720278 EC50 = 0.04 nM T84486 C4KHJ3 118720279 EC50 = 0.05 nM T84486 C85IJS 118720280 EC50 = 0.4 nM T84486 CMK0A4 118720281 EC50 = 0.08 nM T84486 C1KPF5 118720282 EC50 = 0.02 nM T84486 C9XE0M 118720283 EC50 = 0.56 nM T84486 CXV09J 118720284 EC50 = 0.04 nM T84486 C2VF6Q 118720285 EC50 = 0.23 nM T84486 CLE5W1 118720286 EC50 = 0.05 nM T84486 C8QYZ7 118720287 EC50 = 0.78 nM T84486 CMC18U 118720288 EC50 = 0.09 nM T84486 CF1RM4 118720289 EC50 = 0.14 nM T84486 CTS3Q9 118720290 EC50 = 0.3 nM T84486 C8MXV2 118734326 Ki = 0.21 nM T84486 C1G0AS 126705667 EC50 = 0.12 nM T84486 CF1P3M 127048289 Ki = 98.63 nM T84486 CZO71N 127048291 EC50 = 0.47 nM T84486 CI27AJ 127049293 EC50 = 15.57 nM T84486 CE4B3K 127049296 EC50 = 0.59 nM T84486 C92KWB 127049619 EC50 = 14.74 nM T84486 CJ56EF 127049923 EC50 = 0.52 nM T84486 C68PQD 127049995 EC50 > 1000 nM T84486 C0KM6J 127049996 EC50 = 4.23 nM T84486 COZ90D 127049997 EC50 = 2.41 nM T84486 C64VWO 127050537 EC50 > 1000 nM T84486 C31AFY 127051134 EC50 = 283.01 nM T84486 C1S6NE 127051498 EC50 = 0.29 nM T84486 CC8L9I 127051499 EC50 = 7.98 nM T84486 CO75MH 127051770 EC50 = 5.52 nM T84486 C0LM4C 127052688 EC50 = 0.99 nM T84486 C53PTO 127052690 EC50 = 10.79 nM T84486 C2M5AD 127052691 EC50 = 6.98 nM T84486 CA8TZ4 127052735 EC50 = 25.99 nM T84486 CXHF20 127052986 Ki = 6.76 nM T84486 CAG4E0 127052988 EC50 = 4.77 nM T84486 CSP87M 135192889 IC50 = 433 nM T84486 CA6T5H 135192895 IC50 = 223 nM T84486 CC09BD 135192928 IC50 = 30 nM T84486 C2YJ5D 135192930 IC50 = 624 nM T84486 CWQ30S 135192932 IC50 = 9.3 nM T84486 CB8U9O 135192936 IC50 = 23 nM T84486 CM0P9E 135192948 IC50 = 826 nM T84486 CSQ0Y2 135192979 IC50 = 184 nM T84486 CQI48P 135192983 IC50 = 15 nM T84486 CS8A2H 135192997 IC50 = 44 nM T84486 CG3JX8 135193003 IC50 = 235 nM T84486 C7GE0F 135399794 Ki = 448 nM T84486 CHEF49 135399804 Ki > 10000 nM T84486 C1FIH5 135399808 Ki > 10000 nM T84486 CRL41Y 135399831 Ki = 1.6 nM T84486 C86LKI 135413563 EC50 = 28 nM T84486 CK1U7X 135414270 Ki = 174 nM T84486 C8SI4F 135414288 Ki = 61 nM T84486 C9U6OV 135414531 Ki = 3 nM T84486 CVZ9N1 135438362 Ki = 8.7 nM T84486 CO2J1I 135438380 Ki = 36 nM T84486 CMH7K6 135438560 Ki = 15 nM T84486 CXV2S0 135438576 Ki > 214 nM T84486 CD6S8V 135446051 Ki = 37 nM T84486 CS2Z9O 135446053 Ki = 20 nM T84486 CT4GW5 135446078 Ki > 10000 nM T84486 CJ2HL6 135461089 Ki = 6 nM T84486 CYU6R4 135461099 Ki = 21 nM T84486 CCI0M9 135461396 Ki = 322 nM T84486 CFT51M 135466581 Ki = 3.89 nM T84486 CSNQ01 135468119 Ki > 10000 nM T84486 CFS26I 135469685 Ki = 7 nM T84486 CYHQ58 135469700 Ki = 2.089 nM T84486 CK8T6Y 135475778 Ki = 17.78 nM T84486 C0DM8J 135475964 Ki = 60 nM T84486 C3Y5GJ 135475983 Ki > 10000 nM T84486 C4SEV8 135476004 Ki = 0.8913 nM T84486 C3U7PI 135489430 Ki = 109 nM T84486 CTCL26 135491793 Ki = 239 nM T84486 CZK63J 135491819 Ki = 0.9 nM T84486 C9ET1M 135493119 Ki = 1.096 nM T84486 CD53VT 135502557 Ki > 10000 nM T84486 C3W5GY 135505684 Ki > 10000 nM T84486 C59FZN 135505826 Ki > 10000 nM T84486 C0CPM9 135505845 Ki > 10000 nM T84486 CM26GP 135506374 EC50 = 3 nM T84486 C8QL5H 135508167 Ki = 7 nM T84486 CK6S9M 135510027 Ki = 104 nM T84486 CLK7Y3 135513039 Ki = 111 nM T84486 C3DX6C 135515655 Ki = 67 nM T84486 C7P0MW 135520200 Ki = 1376 nM T84486 C8J9EC 135520202 Ki = 18 nM T84486 C4YS7O 135520373 Ki = 64 nM T84486 C5CDZ0 135520376 Ki = 10 nM T84486 CG46WC 135520378 Ki > 10000 nM T84486 CB7S3Y 135530014 Ki = 4.1 nM T84486 CU0WL3 135530164 Ki = 115 nM T84486 CUR82W 135537472 Ki = 67 nM T84486 CRY3M0 135613341 Ki = 237 nM T84486 CY12JN 135644174 Ki = 4900 nM T84486 CT0A1P 135916059 Ki = 111 nM T84486 CHJ03T 135916060 Ki > 1000 nM T84486 CO6G5W 135916061 Ki > 5000 nM T84486 C5T1NJ 135916062 Ki > 5000 nM T84486 CAN9M3 135916069 Ki = 27.8 nM T84486 CH2L4N 135916070 Ki = 17 nM T84486 C32QZC 135997467 Ki = 1750 nM T84486 CO03UG 136961690 Ki = 6.22 nM T84486 CYA2L4 137189941 Ki > 10000 nM T84486 CY64JO 137212769 Ki > 10000 nM T84486 CY3E7O 137212770 Ki = 7452 nM T84486 C1YN5T 137212771 Ki > 10000 nM T84486 CI0HQ6 137212772 Ki = 801 nM T84486 C0U2ZG 137212773 Ki > 10000 nM T84486 C81USM 137212774 Ki > 10000 nM T84486 CHZM41 137212775 Ki > 10000 nM T84486 CD2SQ5 137212776 Ki = 8349 nM T84486 CNZR50 137631348 EC50 = 0.11 nM T84486 CSKL70 137632034 EC50 = 0.027 nM T84486 CON47G 137632998 EC50 = 0.0072 nM T84486 CWJO17 137633699 EC50 > 100 nM T84486 CTNY20 137634089 EC50 = 0.082 nM T84486 CGZ12O 137634607 EC50 = 0.056 nM T84486 C0JLD1 137635522 EC50 = 1.2 nM T84486 CTK80A 137635922 EC50 = 1.6 nM T84486 C73GYS 137636048 EC50 > 100 nM T84486 CO2Q1A 137637782 EC50 = 4.4 nM T84486 CU6F1L 137638040 EC50 = 1.5 nM T84486 CW2FA1 137639236 EC50 = 0.11 nM T84486 CGHQ73 137639317 EC50 > 100 nM T84486 CKSY39 137639340 EC50 = 0.26 nM T84486 CS1D6A 137639396 EC50 = 0.007 nM T84486 CD5C8H 137640536 EC50 > 100 nM T84486 CH8DK2 137640630 EC50 = 3.4 nM T84486 CEWQ40 137641012 EC50 = 0.25 nM T84486 C8TNJ3 137641033 EC50 = 0.0086 nM T84486 CNKR47 137643372 EC50 = 1.4 nM T84486 C1NYP7 137645401 EC50 = 0.014 nM T84486 CD3NB0 137646127 EC50 > 100 nM T84486 C0IVK7 137647081 EC50 > 100 nM T84486 CNZ60A 137647351 EC50 = 0.042 nM T84486 CO6DZ8 137647481 EC50 = 1.6 nM T84486 CFG78N 137648249 EC50 = 5.1 nM T84486 CM5SI7 137648427 EC50 = 0.19 nM T84486 C92UGK 137648677 EC50 = 0.054 nM T84486 C61EOM 137649234 EC50 = 0.12 nM T84486 CMS7U4 137650792 EC50 = 0.015 nM T84486 C34LGF 137651105 EC50 = 0.0055 nM T84486 C94TRJ 137651797 EC50 = 22 nM T84486 CBC95F 137652261 EC50 = 89 nM T84486 CI0QE4 137652597 EC50 = 0.03 nM T84486 C41YXQ 137652984 EC50 = 0.19 nM T84486 C0AT6R 137653368 EC50 > 100 nM T84486 C2TW5S 137653639 EC50 = 0.021 nM T84486 CIF85C 137653770 EC50 = 9.5 nM T84486 CL9YJ6 137653847 EC50 = 0.013 nM T84486 CW8G3A 137654006 EC50 = 0.013 nM T84486 CK73UR 137654009 EC50 = 0.78 nM T84486 CG1DK7 137654217 EC50 = 0.031 nM T84486 C2N3TK 137654636 EC50 = 40 nM T84486 CVS36J 137654665 EC50 = 0.35 nM T84486 C3PSE5 137654909 EC50 > 100 nM T84486 CWN2I1 137654919 EC50 = 0.12 nM T84486 CB20TQ 137656338 EC50 = 0.0069 nM T84486 CAZL21 137656718 EC50 = 3.6 nM T84486 C3NM6I 137657345 EC50 = 0.0075 nM T84486 CB6FS3 137658004 EC50 = 17 nM T84486 C0C7MG 137658241 EC50 = 12 nM T84486 CWI56Q 137658998 EC50 = 0.0053 nM T84486 CKR3T2 137659747 EC50 = 0.53 nM T84486 C56UYT 137659822 EC50 = 0.24 nM T84486 CH19JW 137660341 EC50 = 0.01 nM T84486 C9EDO4 137660579 EC50 = 0.0065 nM T84486 C5EU8T 137661047 EC50 = 0.027 nM T84486 C5V6BP 137661245 EC50 = 0.072 nM T84486 CZ7FL0 137662128 EC50 > 100 nM T84486 CT5D3X 142391767 IC50 = 132 nM T84486 CTO5N4 142391805 IC50 = 52 nM T84486 C7XTV3 145711714 EC50 = 25 nM T84486 C6ZU0A 145949555 IC50 > 20000 nM T84486 CIY9U2 145949926 IC50 > 10000 nM T84486 C5INL8 145950135 Ki > 10000 nM T84486 CE3D8P 145951877 IC50 > 20000 nM T84486 CI9BO4 145952624 IC50 = 5320 nM T84486 CL42TO 145953024 IC50 = 6780 nM T84486 C9XH8D 145953061 IC50 > 10000 nM T84486 CF5I1P 145953063 Ki > 10000 nM T84486 CS4FG6 145955181 Ki > 10000 nM T84486 C14WVM 145956003 IC50 > 10000 nM T84486 C5C8IL 145956239 Ki > 10000 nM T84486 CR2QH0 145957924 IC50 = 5760 nM T84486 CP25CA 145958767 IC50 > 20000 nM T84486 C6F0CS 145959206 Ki > 10000 nM T84486 C6AVU4 145959208 Ki > 10000 nM T84486 C3Z9BN 145959348 Ki > 10000 nM T84486 CBP35Y 145959434 Ki > 10000 nM T84486 C63UNT 145960494 EC50 = 109 nM T84486 CIG1P6 145961670 Ki = 166 nM T84486 C53JQB 145962220 EC50 = 34 nM T84486 CRXH51 145963213 Ki = 220 nM T84486 CB3TK5 145964151 EC50 = 6.8 nM T84486 CY0FL4 145964296 Ki = 340 nM T84486 C9U4FR 145964703 EC50 = 0.44 nM T84486 CS40EH 145965644 Ki < 10 nM T84486 CYSP85 145965794 Ki = 385 nM T84486 CAHB80 145966126 Ki > 1000 nM T84486 C3R0NB 145966470 EC50 = 0.77 nM T84486 CTC9Q6 145966784 EC50 = 0.6 nM T84486 CYIE13 145970269 Ki = 417 nM T84486 C3H7SY 145970757 Ki = 37.4 nM T84486 CLN68K 145971236 Ki > 10000 nM T84486 C43AQD 145971417 Ki = 1333 nM T84486 C01GKQ 145971455 IC50 > 20000 nM T84486 CJF16G 145972114 EC50 = 300 nM T84486 CPY61F 145972843 Ki < 10 nM T84486 CK8HA2 145973088 EC50 = 28 nM T84486 CI9G0B 145974527 Ki = 61 nM T84486 CFQ05K 145974615 Ki < 10 nM T84486 CNF1J3 145974638 Ki = 686 nM T84486 C7P6YW 145974697 EC50 = 0.83 nM T84486 CXD4H3 145974945 EC50 = 194 nM T84486 CY2MW6 145975112 EC50 = 0.51 nM T84486 CVE64Z 145975166 Ki = 150 nM T84486 CQB98S 145975622 EC50 = 3.6 nM T84486 C3XM4U 145975847 EC50 = 5.2 nM T84486 CJT06P 145976546 Ki = 800 nM T84486 CQ2IG7 145976595 IC50 = 37 nM T84486 CF14DJ 145976648 Ki = 104 nM T84486 C4B3WF 145976821 EC50 = 1.3 nM T84486 C15KIT 145977344 EC50 = 1.8 nM T84486 CS5CD6 145977918 Ki > 1000 nM T84486 C8K1EH 145977939 EC50 = 5.4 nM T84486 CX16OC 145978563 EC50 = 0.6 nM T84486 CT1PI4 145978570 Ki = 84 nM T84486 CTYI46 145978612 Ki < 10 nM T84486 CK83JH 145978698 EC50 = 1.8 nM T84486 C0IC1N 146238444 IC50 = 27 nM T84486 CS3L9V 155515303 EC50 = 10.47 nM T84486 CSB84H 155515636 EC50 > 100000 nM T84486 C9IX5T 155516256 IC50 = 1227 nM T84486 C57MKA 155517601 IC50 = 121 nM T84486 CI4T0F 155518894 EC50 > 100000 nM T84486 CPA8S4 155520603 IC50 = 10 nM T84486 C8BKV3 155523986 EC50 = 160 nM T84486 CDN37P 155524296 EC50 > 100000 nM T84486 C1MFP0 155524463 EC50 = 65.49 nM T84486 C2RPD0 155527198 EC50 = 0.089 nM T84486 CY1A5R 155527834 EC50 = 4.8 nM T84486 CA75ZF 155527876 EC50 > 100000 nM T84486 CT8L7Z 155529697 EC50 = 5.28 nM T84486 CYOF34 155532160 EC50 = 0.15 nM T84486 C8OT1G 155533728 EC50 > 10000 nM T84486 C4ZC5Y 155536940 EC50 = 0.028 nM T84486 C2DFI0 155537980 IC50 = 6759 nM T84486 CT41UO 155542139 IC50 = 1379 nM T84486 CK1M8N 155542151 EC50 = 0.0012 nM T84486 CT80FD 155542264 EC50 = 0.0008 nM T84486 CA6DC4 155542670 EC50 > 10000 nM T84486 CWO69R 155547112 EC50 > 1000 nM T84486 C8YZU4 155547725 EC50 = 4.1 nM T84486 C7N8YM 155548766 EC50 = 2.58 nM T84486 CU5SX6 155551252 EC50 = 0.00257 nM T84486 CJSW73 155551624 EC50 > 1000 nM T84486 C9EBM8 155552392 EC50 = 3.41 nM T84486 CGS75B 155553462 EC50 = 11.78 nM T84486 CMC53Q 155553492 EC50 = 5.27 nM T84486 C6NRL8 155554422 IC50 = 2794 nM T84486 C2JH0F 155555127 EC50 = 20.7 nM T84486 CSA2B9 155555256 EC50 = 14.42 nM T84486 C7Q8AH 155558305 IC50 = 2561 nM T84486 CL93EY 155558494 EC50 = 52.44 nM T84486 CH5V4G 155559767 EC50 = 0.265 nM T84486 CY97OP 155560248 EC50 = 0.0014 nM T84486 C0HLS3 155564470 IC50 = 401 nM T84486 CJVC24 155565553 IC50 = 910 nM T84486 COX4M3 155565903 EC50 = 0.031 nM T84486 C5RJ2L 155568614 IC50 = 850 nM T84486 C6MQS7 155569305 EC50 > 1000 nM T84486 D00SGZ 9917025 Ki = 71 nM T84486 D01EDA 44429298 IC50 = 40 nM T84486 D01WHI 135413562 Ki = 0.65 nM T84486 D06SMJ 44429300 IC50 = 7850 nM T84486 D07HTH 44429290 IC50 = 51 nM T84486 D07KWZ 10413997 Ki = 61 nM T84486 D07NPZ 44429299 IC50 = 1002 nM T84486 D07XKF 16737617 IC50 = 103 nM T84486 D08MTW 44429250 IC50 = 7 nM T84486 D09LXI 44429294 IC50 = 25 nM T84486 D09RIE 44419028 Ki = 240 nM T84486 D0F9QJ 44429264 IC50 = 1380 nM T84486 D0H0MK 44429303 IC50 = 485 nM T84486 D0I3HV 44429288 IC50 = 176 nM T84486 D0IB4H 16737618 IC50 = 380 nM T84486 D0K5NV 44428109 Ki = 1.95 nM T84486 D0L0RP 44428107 Ki = 1.04 nM T84486 D0NC8V 6918854 Ki = 1.259 nM T84486 D0O1KA 16737793 IC50 = 75 nM T84486 D0O9FA 44429304 IC50 = 55 nM T84486 D0Q0OR 10461270 Ki = 0.5 nM T84486 D0R1WH 16738355 IC50 = 130 nM T84486 D0R7QC 44419039 Ki = 1083 nM T84486 D0S3GE 16738356 IC50 = 730 nM T84486 D0T4ML 5311202 Ki = 4.1 nM T84486 D0W3IQ 44419025 Ki = 136 nM T84486 D0Y0SO 44419026 EC50 = 350 nM T84486 D0YG0D 9797987 Ki = 1000 nM T84486 D0YL6T 16736614 IC50 = 8500 nM T84486 D0ZD0W 11366713 Ki = 326 nM T84486 D0ZV3Y 44429295 IC50 = 80 nM T44150 D0R9YR 64971 EC50 > 50000 nM T44150 CD96MY 10553584 EC50 > 50000 nM T44150 C0C6KD 11190936 EC50 > 50000 nM T44150 CO7Z5W 21671980 EC50 > 50000 nM T44150 C7NB9R 127037042 EC50 = 16400 nM T44150 CINW82 127037404 EC50 = 7700 nM T44150 C2O9ES 134437859 EC50 = 11400 nM T44150 CD1RN6 134437860 EC50 = 3800 nM T44150 CDT1G2 134437890 EC50 = 5000 nM T44150 C5OJA3 134437938 EC50 = 7100 nM T44150 C4U6VF 155511857 EC50 = 8900 nM T44150 C4M3QA 155527583 EC50 = 3200 nM T44150 C8T1QA 155529758 EC50 = 2400 nM T44150 C5B2QV 155530595 EC50 = 2600 nM T44150 C7T8LF 155535380 EC50 = 5800 nM T44150 CCN2K1 155536446 EC50 > 50000 nM T44150 C84BEX 155539396 EC50 = 4800 nM T44150 CB1KZ4 155561830 EC50 = 6800 nM T44150 CQPR47 155569312 EC50 = 7500 nM T44150 D01BZE 73659 EC50 > 50000 nM T44150 D07LUJ 64945 EC50 > 50000 nM T44150 D0SJ2Q 10494 EC50 > 50000 nM T44150 D0U8IF 10114 EC50 > 50000 nM T99616 D0ZS8P 2801 IC50 = 3400 nM T99616 CT48KR 21025 IC50 = 11800 nM T99616 CQ89PJ 69920 IC50 = 9300 nM T99616 CCZ04P 214232 IC50 = 7800 nM T99616 C8MEI0 223143 IC50 = 340 nM T99616 CJKN12 432139 IC50 = 3300 nM T99616 CN1TR3 580286 IC50 = 3300 nM T99616 C39UQA 723918 IC50 = 148000 nM T99616 CTX3F0 831028 IC50 = 107000 nM T99616 C2ZL6W 877340 IC50 = 1500 nM T99616 CV0S1M 877450 IC50 = 1700 nM T99616 CD4IA9 1712537 IC50 = 38800 nM T99616 CK1N3W 2223018 IC50 = 2400 nM T99616 C2O8ZG 2288440 IC50 = 2000 nM T99616 CG5CX3 2857821 IC50 = 37000 nM T99616 C1ESQ4 2862129 IC50 = 6800 nM T99616 CJ50SW 2862130 IC50 = 23000 nM T99616 C1AL8J 2870196 IC50 = 15000 nM T99616 CM86QC 2870319 IC50 = 67000 nM T99616 CQ4W7L 2870365 IC50 > 100000 nM T99616 CO1XP5 2870470 IC50 = 89000 nM T99616 CFJR69 2874741 IC50 = 37000 nM T99616 CW26DB 2874772 IC50 = 12000 nM T99616 C86JXI 2926799 IC50 = 9400 nM T99616 CU9IK5 3117554 IC50 > 100000 nM T99616 C0SZ5P 3119180 IC50 = 93000 nM T99616 CKNP81 3123254 IC50 > 100000 nM T99616 CZ87AQ 3304561 IC50 > 100000 nM T99616 CI41EX 3515999 IC50 = 39000 nM T99616 CSZU71 4448737 IC50 = 2900 nM T99616 CIEG57 10632580 IC50 = 69200 nM T99616 C71CVZ 10803696 IC50 = 7600 nM T99616 C6D0LI 23644650 IC50 = 870 nM T99616 CCFM84 53252998 IC50 = 4880 nM T99616 C3Q4ET 54669774 Ki = 190 nM T99616 CS8O6N 54756882 IC50 = 710 nM T99616 C8XYW1 54756883 IC50 = 730 nM T99616 C8ZCJ9 54756884 IC50 = 4900 nM T99616 CU1F4I 54756885 IC50 = 1500 nM T99616 C3AB7M 54756886 IC50 = 590 nM T99616 C5ULB0 54756887 IC50 = 1200 nM T99616 CRT20Z 54756888 IC50 = 4600 nM T99616 CLA79P 54756986 IC50 = 4900 nM T99616 CN3BC1 54756987 IC50 = 6800 nM T99616 CFBI15 54757489 IC50 = 53000 nM T99616 C6PWG5 54757490 IC50 = 24000 nM T99616 CZP7R4 54757592 IC50 = 1700 nM T99616 CF7O3K 54757594 IC50 = 50000 nM T99616 CZ91FK 54757595 IC50 = 20000 nM T99616 CAN47L 54757596 IC50 = 1600 nM T99616 CV87KH 54757706 IC50 = 930 nM T99616 C78NDU 54757707 IC50 = 2000 nM T99616 CZE1U4 54757708 IC50 = 1100 nM T99616 C6XW8O 54757709 IC50 = 940 nM T99616 C4V2IL 54757710 IC50 = 3500 nM T99616 CQC39N 54757711 IC50 = 1500 nM T99616 CBOP24 54757712 IC50 = 810 nM T99616 CL0KS4 54757801 IC50 = 1300 nM T99616 C9PQ8X 54757802 IC50 = 2200 nM T99616 CSCY30 54757803 IC50 = 2200 nM T99616 CHJ64V 54757804 IC50 = 1200 nM T99616 C67YLS 54757805 IC50 = 1800 nM T99616 C92JDY 54757806 IC50 = 2800 nM T99616 CG2HB7 54757807 Ki = 320 nM T99616 CB81DI 54757897 IC50 = 3500 nM T99616 C8ZAP2 54757898 IC50 = 1000 nM T99616 C90XFK 54757899 IC50 = 2000 nM T99616 CW4I8S 54757900 IC50 = 2600 nM T99616 CE3BM6 54757901 IC50 = 2100 nM T99616 CTBA16 54757902 IC50 = 2300 nM T99616 C5C7QB 54757903 IC50 = 1700 nM T99616 C62BNH 54757996 Ki = 440 nM T99616 CYZ4B5 54757997 IC50 = 1800 nM T99616 CPJ95H 54757998 IC50 = 1300 nM T99616 CVH3I9 54757999 IC50 = 810 nM T99616 CJEF45 54758000 IC50 = 1500 nM T99616 C1JLY6 54758001 IC50 = 1700 nM T99616 C6B4OX 54758091 IC50 = 1500 nM T99616 C35AYN 54758092 IC50 = 1600 nM T99616 CKGA16 54758093 IC50 = 420 nM T99616 CY03OS 54758094 IC50 = 2000 nM T99616 CH6VS8 54758095 IC50 = 1600 nM T99616 C0HV6O 54758096 Ki = 270 nM T99616 C5O2FP 54758181 IC50 = 780 nM T99616 C19WVD 54758182 IC50 = 790 nM T99616 CB0TJ1 54758183 IC50 = 350 nM T99616 CM1QX5 54758184 IC50 = 7300 nM T99616 C39ODN 54758185 IC50 = 4400 nM T99616 CS0X6J 54758186 IC50 = 1300 nM T99616 CU7W6H 54758274 IC50 = 790 nM T99616 C0KN6G 54758275 IC50 = 8000 nM T99616 CJE27G 54758276 IC50 = 8500 nM T99616 CJZ7K0 54758370 IC50 = 7900 nM T99616 COEZ47 54758371 IC50 = 900 nM T99616 CM5PF9 54758372 IC50 = 28000 nM T99616 CVT01Z 54758373 IC50 = 1300 nM T99616 C6PU4F 54758374 IC50 = 27000 nM T99616 CW7P2U 54758375 IC50 = 8300 nM T99616 C72JWG 71455461 Ki = 3400 nM T99616 CD7JB2 71462602 Ki = 2800 nM T99616 C9R8BW 122184261 IC50 = 7390 nM T99616 C9M7NF 127026790 IC50 = 7200 nM T99616 C2ZKR3 145983314 Ki = 7500 nM T99616 D00DKI 10107976 IC50 = 5000 nM T25703 CFX34A 11624321 IC50 = 1500 nM T25703 CNBJ09 25141638 IC50 = 2600 nM T25703 CL2Q6J 44178077 IC50 = 1900 nM T25703 CVF83A 57775660 IC50 = 250 nM T25703 C2KJ3Q 58580498 IC50 = 60 nM T25703 CYN1P7 71421283 IC50 = 900 nM T25703 C1TPZ2 155515265 IC50 = 54000 nM T76846 D0H7AR 70684954 Ki = 68000 nM T76846 D0LI1C 44469321 IC50 > 30000 nM T76846 D0X9PF 9941379 EC50 = 2.399 nM T76846 CL04VQ 910537 Ki > 1000000 nM T76846 C0DA9X 2163781 Ki = 86000 nM T76846 CK4YT2 2817655 Ki > 1000000 nM T76846 CB9A2M 2852098 Ki = 59000 nM T76846 C8EPT1 6918707 IC50 = 280 nM T76846 CWZ1O2 6918780 EC50 > 10000 nM T76846 CY60AZ 6918813 EC50 = 990 nM T76846 C2BQE1 6918814 Ki = 640 nM T76846 CK83QR 6918844 Ki = 790 nM T76846 CLV3C7 6918849 IC50 = 32 nM T76846 C5U7CS 6918850 Ki = 1100 nM T76846 C0Q5JL 6918851 IC50 = 942 nM T76846 CRG04O 6918857 Ki = 7000 nM T76846 COS6C1 9808720 EC50 > 10000 nM T76846 CM02VS 9808801 IC50 = 230 nM T76846 CY4K7X 9849434 EC50 = 148 nM T76846 CKCF18 9867330 EC50 = 230 nM T76846 CM3Y5H 9893728 IC50 > 10000 nM T76846 CZ5E2C 9915636 Ki = 1000 nM T76846 C15DES 9924916 Ki = 68000 nM T76846 C7V8AE 9946241 Ki = 16000 nM T76846 C6L4VG 9946358 Ki = 127000 nM T76846 CX5CU3 9958649 Ki = 3900 nM T76846 C97MRJ 9960253 EC50 = 2000 nM T76846 CMU31X 9968756 Ki = 29000 nM T76846 C5F3QU 9969456 Ki = 19000 nM T76846 CLXA58 10025669 Ki = 50118.72 nM T76846 CRP4X1 10030530 IC50 > 10000 nM T76846 CZ78WX 10077258 EC50 = 1800 nM T76846 C8MCA1 10077773 Ki = 400 nM T76846 CSQ60B 10108894 Ki = 14000 nM T76846 C6LVA2 10109225 Ki = 17000 nM T76846 CG1K8Y 10122170 EC50 > 10000 nM T76846 CF81WV 10132207 Ki = 134000 nM T76846 C0PVS9 10134057 Ki = 9100 nM T76846 CC0ZT7 10137615 Ki = 12000 nM T76846 CO69QN 10146211 EC50 = 7000 nM T76846 C03AKT 10155513 Ki = 44000 nM T76846 CPRS08 10157774 Ki = 50000 nM T76846 CXF16O 10158674 Ki = 58000 nM T76846 C97IHD 10159196 Ki = 38000 nM T76846 CAB06U 10177247 Ki = 63000 nM T76846 COJ1M5 10178845 Ki = 7400 nM T76846 CV2QX0 10180932 Ki = 20000 nM T76846 C78FGS 10188529 IC50 = 1350 nM T76846 C1HMR6 10200110 Ki = 63000 nM T76846 CFZ5I6 10210964 IC50 = 83 nM T76846 C8PA3J 10211466 Ki = 16000 nM T76846 CWJ5I0 10225762 Ki = 33000 nM T76846 CTO7I8 10232787 Ki = 3400 nM T76846 CSNY06 10257242 EC50 = 2000 nM T76846 C6Y1ER 10257541 Ki = 4400 nM T76846 C2AL7S 10260053 EC50 = 68 nM T76846 CEC2M0 10269187 Ki = 131000 nM T76846 C6T2MU 10270570 Ki = 11000 nM T76846 CX29KB 10282847 IC50 = 170 nM T76846 C4SCW2 10283036 Ki = 1900 nM T76846 C01QVJ 10291369 Ki = 21000 nM T76846 CSDX25 10291370 Ki = 24000 nM T76846 CX97KY 10292084 Ki = 37000 nM T76846 CU17RB 10293285 Ki = 12000 nM T76846 CV3ZJ5 10304463 Ki = 1400 nM T76846 CU13DH 10304547 IC50 = 120 nM T76846 C1E3PC 10304776 IC50 = 97 nM T76846 CT9AR6 10325955 EC50 = 1600 nM T76846 C1N3MA 10392968 IC50 = 48000 nM T76846 CPL02I 10463896 EC50 = 136.4 nM T76846 CTEB92 10483153 IC50 = 970 nM T76846 C3NWO8 10484741 EC50 = 170 nM T76846 CGIC31 10918643 IC50 > 10000 nM T76846 C7IJV5 11038873 EC50 = 1700 nM T76846 CHOS10 11061068 EC50 = 59 nM T76846 CO2U6S 11156852 Ki = 33 nM T76846 C3V7DK 11180881 Ki = 1400 nM T76846 CHC51K 11181804 Ki = 1800 nM T76846 CDLG18 11205265 EC50 = 6309.57 nM T76846 C9WTR4 11205266 IC50 = 1258.93 nM T76846 CDMB38 11205293 EC50 = 6309.57 nM T76846 CD5SG6 11215758 Ki = 630 nM T76846 CF7VQ4 11226756 EC50 = 1800 nM T76846 CWLJ34 11237444 Ki = 2400 nM T76846 C1T3VM 11249545 Ki = 2800 nM T76846 C6FBD3 11251566 EC50 = 316.23 nM T76846 C6ETW3 11251567 EC50 = 5011.87 nM T76846 C9LOV4 11251591 IC50 = 3981.07 nM T76846 CMI4E5 11251592 EC50 = 158.49 nM T76846 C0D1PE 11263072 EC50 = 25.12 nM T76846 CP9S6F 11273288 EC50 = 150 nM T76846 C07VJD 11274575 EC50 = 501.19 nM T76846 CJ7OT2 11296600 Ki = 2000 nM T76846 C2PU1F 11296732 Ki = 1900 nM T76846 CYH1I3 11297620 IC50 = 44 nM T76846 C9XBQ7 11308054 Ki = 258 nM T76846 C97ICV 11309021 IC50 = 1995.26 nM T76846 CVE6D9 11309022 EC50 = 5011.87 nM T76846 CS7K4R 11341045 Ki = 2200 nM T76846 CU6Y1Z 11341046 Ki = 2500 nM T76846 CAL3F9 11364326 Ki = 2800 nM T76846 CEX40J 11366515 EC50 = 794.33 nM T76846 C5D1TY 11375764 Ki = 3500 nM T76846 CR8B4G 11378033 EC50 = 3162.28 nM T76846 CQ1ZL6 11411962 EC50 = 3981.07 nM T76846 CUTZ31 11445925 EC50 = 3981.07 nM T76846 C2DNI1 11468666 EC50 = 630.96 nM T76846 C8LN5W 11477853 Ki = 2300 nM T76846 CVR0T4 11490658 Ki = 1900 nM T76846 CH7TQ6 11753695 EC50 = 351 nM T76846 CUL54T 11764499 EC50 = 158.49 nM T76846 C2SHV7 11786860 Ki = 3600 nM T76846 CD9N5B 11787842 IC50 = 7943.28 nM T76846 CQ06HS 11787864 EC50 = 1995.26 nM T76846 C0OIV9 11813437 EC50 = 7000 nM T76846 C7NL4J 11845272 Ki = 86 nM T76846 C4XF1I 11845276 Ki = 403 nM T76846 CT1F9R 11845438 EC50 = 825 nM T76846 CC42HM 11845440 EC50 = 2474 nM T76846 CFKN79 11845444 Ki = 19213 nM T76846 C3JV7M 11845450 EC50 = 1.3 nM T76846 C8WJ6E 11845630 EC50 = 1171 nM T76846 CI1VU0 11845804 EC50 = 3720 nM T76846 C4V9DO 11845813 EC50 = 871 nM T76846 CSZX65 11846669 Ki = 156 nM T76846 C5HFB2 11846673 Ki = 289 nM T76846 C25KCW 11846844 EC50 = 68 nM T76846 CO3H9V 11847001 EC50 = 1134 nM T76846 CECQ63 11847312 EC50 = 1774 nM T76846 CT4EC3 11966875 IC50 > 10000 nM T76846 CI9W3G 15953833 IC50 = 420 nM T76846 CAT74W 15953838 IC50 = 2172 nM T76846 C2BLT4 16007263 EC50 = 41 nM T76846 C54MIL 16007264 Ki = 1200 nM T76846 C6XS3N 16007285 Ki = 800 nM T76846 CYW0B8 16038315 Ki = 5000 nM T76846 C4N0VF 16046215 Ki = 1300 nM T76846 CX68DN 16049796 EC50 > 10000 nM T76846 C8UXP9 16126683 EC50 = 350 nM T76846 CPTO16 16132144 EC50 = 0.669 nM T76846 C4NZ3C 16725559 IC50 = 4293 nM T76846 C25XZF 17880880 Ki > 1000000 nM T76846 CFNQ06 23635107 Ki = 230 nM T76846 CHU29W 23635235 Ki = 420 nM T76846 CWL5K4 23635236 Ki = 710 nM T76846 CVFQ41 23635237 Ki = 270 nM T76846 CBW09O 23653113 Ki = 53000 nM T76846 C8KO9M 23661656 Ki = 1800 nM T76846 CK2Q5J 24180592 Ki = 710 nM T76846 C7SMW5 24180646 Ki = 750 nM T76846 CU19BT 24740419 Ki = 3300 nM T76846 CTC05L 24740653 Ki = 2800 nM T76846 CD90WZ 24740655 Ki = 820 nM T76846 CUPD43 24741624 Ki = 320 nM T76846 C5TA3W 24774358 EC50 = 100 nM T76846 CO4JK2 24774437 IC50 > 10000 nM T76846 CMB27G 24774521 IC50 = 20 nM T76846 C2TAK6 24774601 IC50 > 1000 nM T76846 C2A1SX 24848995 Ki = 24 nM T76846 C1EN7W 24857886 IC50 = 3777 nM T76846 CJZ5U2 24858922 IC50 > 1000 nM T76846 CB9M3F 24873537 Ki = 1600 nM T76846 CS0L2N 24882666 Ki = 3500 nM T76846 CG9AV5 25058412 Ki = 1700 nM T76846 CJ5HN6 25128748 EC50 = 300 nM T76846 C3WE0T 25128749 EC50 = 113 nM T76846 CP5TN2 25128751 Ki = 428 nM T76846 CUTA14 25129105 Ki = 144 nM T76846 CPL49Z 25129107 EC50 = 44 nM T76846 C4N5DH 25129108 EC50 = 58 nM T76846 CDC2Q6 25129109 EC50 = 51 nM T76846 CVSO97 25129453 EC50 = 12 nM T76846 CE79VX 25131477 Ki = 26323 nM T76846 C1B7KF 25131478 Ki = 76 nM T76846 CIJ6P4 25132524 EC50 = 237 nM T76846 CY42MT 25132525 EC50 = 271 nM T76846 C9QG3J 25132526 EC50 = 545 nM T76846 CL3JV6 25132864 Ki = 170 nM T76846 C57QZT 25132866 EC50 = 103 nM T76846 CR6YZ2 25132867 Ki = 215 nM T76846 C8AO5Y 25133207 Ki = 434 nM T76846 C3VGX6 25133208 EC50 = 84 nM T76846 C3KRA8 25133209 EC50 = 52 nM T76846 C9U6CQ 25133210 EC50 = 40 nM T76846 C74ACT 25133556 EC50 = 108 nM T76846 CW7O1N 25133903 Ki = 8734 nM T76846 CG3R0Y 25133907 EC50 = 149 nM T76846 C4SH1P 25211670 Ki = 3100 nM T76846 C4HK6C 42630327 EC50 = 0.6918 nM T76846 CIOF26 44158168 IC50 = 1 nM T76846 C53LJK 44158169 EC50 = 2500 nM T76846 C9UD8I 44158336 EC50 = 620 nM T76846 CF6PT4 44158337 EC50 = 130 nM T76846 CHKI60 44265225 Ki > 1000000 nM T76846 CXN2R4 44265309 Ki = 57000 nM T76846 C3EJ1R 44265312 Ki = 214000 nM T76846 CWPT03 44265315 Ki = 167000 nM T76846 CJ1M6N 44265347 Ki = 58000 nM T76846 CEQ6K7 44265351 Ki = 294000 nM T76846 CSL48C 44265374 Ki = 33000 nM T76846 C97AIK 44265472 Ki = 45000 nM T76846 CLE96R 44265479 Ki > 1000000 nM T76846 CV8GX6 44265487 Ki = 31000 nM T76846 C2CPG9 44265489 Ki = 145000 nM T76846 CLP5G3 44265496 Ki = 7943.28 nM T76846 C51TPY 44265586 Ki > 1000 nM T76846 CH5WM7 44265588 Ki > 1000 nM T76846 CT89LY 44265589 Ki = 107000 nM T76846 CZS3C7 44265590 Ki = 155000 nM T76846 C3YKG9 44265591 Ki = 147000 nM T76846 C74SBD 44265625 Ki > 1000 nM T76846 CRQ92O 44265626 Ki > 1000 nM T76846 CT2S8I 44265639 Ki = 6400 nM T76846 C18JZD 44265656 Ki > 1000000 nM T76846 CD8UC0 44265662 Ki > 1000 nM T76846 C6OU7D 44265665 Ki > 1000 nM T76846 CC28FH 44265672 Ki = 37000 nM T76846 CSK9V6 44265674 Ki > 1000 nM T76846 CS46LN 44265675 Ki > 1000000 nM T76846 C9E0TB 44265681 Ki = 82000 nM T76846 CCGI15 44265707 Ki = 28000 nM T76846 CION54 44265708 Ki > 1000000 nM T76846 C9CM8W 44265711 Ki = 53000 nM T76846 CPUO61 44265713 Ki = 161000 nM T76846 CP1E6X 44265715 Ki = 14000 nM T76846 CRFQ64 44265719 Ki > 1000000 nM T76846 CXUI50 44265722 Ki = 161000 nM T76846 CVEG42 44265727 Ki > 1000 nM T76846 CC4S8V 44265739 Ki > 1000 nM T76846 CG1CH0 44265748 Ki > 1000 nM T76846 C82FPN 44265749 Ki = 56000 nM T76846 C05MIH 44265751 Ki = 4800 nM T76846 CP82FI 44265757 Ki > 1000 nM T76846 CE6A0Z 44265759 Ki > 1000 nM T76846 CPE83Q 44269189 EC50 = 2200 nM T76846 CCP5L2 44269214 EC50 = 3900 nM T76846 CN5TI2 44269217 EC50 = 250 nM T76846 CBW0I1 44275650 EC50 = 6 nM T76846 C5OHC4 44277696 IC50 = 4000 nM T76846 CU8PH5 44293516 EC50 = 88.5 nM T76846 C7DZ1Q 44293599 IC50 > 1000 nM T76846 C57HNX 44307979 IC50 > 10000 nM T76846 C8LZV7 44308004 IC50 > 10000 nM T76846 CFP7W8 44308044 IC50 > 10000 nM T76846 C79WRA 44308214 IC50 > 10000 nM T76846 CT76SR 44308215 IC50 > 10000 nM T76846 COY71H 44314826 IC50 = 23 nM T76846 CJAW38 44314951 IC50 > 10000 nM T76846 CA7B1G 44315095 IC50 = 10000 nM T76846 CPX2L1 44315335 IC50 > 10000 nM T76846 CQ59BO 44320339 Ki = 31622.78 nM T76846 C6UML0 44322786 EC50 = 840 nM T76846 C3CL8S 44322787 EC50 = 40.5 nM T76846 C5SZ6K 44322788 EC50 = 450 nM T76846 C27QTD 44322795 EC50 = 70 nM T76846 C9HQ8Z 44322812 EC50 = 71 nM T76846 C3XED9 44322868 Ki = 5.9 nM T76846 C8P1HE 44322869 EC50 = 75 nM T76846 CJD5K7 44322895 EC50 = 6 nM T76846 CSH73B 44322896 EC50 = 4.7 nM T76846 C3V7PO 44322923 EC50 = 160 nM T76846 CA9F8I 44322924 EC50 = 300 nM T76846 C32ADM 44322957 EC50 = 120 nM T76846 CU1R6F 44322958 EC50 = 13 nM T76846 CPG80V 44322959 EC50 = 45 nM T76846 CJ73UR 44322977 EC50 = 58 nM T76846 CW5T8L 44322986 EC50 = 130 nM T76846 CN12SY 44322987 EC50 = 93.3 nM T76846 C8W2GN 44322994 Ki = 380 nM T76846 CEV0F8 44323015 Ki = 230 nM T76846 CSL38N 44323016 EC50 = 390 nM T76846 CEDS20 44323020 Ki = 7.8 nM T76846 CI70FV 44323029 EC50 = 9.3 nM T76846 CNB32J 44323031 EC50 = 17 nM T76846 CP9FE1 44323032 EC50 = 28 nM T76846 CCX5N0 44323033 EC50 = 98.3 nM T76846 C7RT2W 44323034 Ki = 440 nM T76846 CTQI30 44323211 Ki = 370 nM T76846 CC9E1M 44323212 Ki = 1400 nM T76846 CX7H2C 44323233 EC50 = 13 nM T76846 CW49BO 44323234 Ki = 12.1 nM T76846 C8BID0 44325926 IC50 = 50.04 nM T76846 C9MA4R 44343337 EC50 = 0.191 nM T76846 CD9ER8 44343341 EC50 = 2.813 nM T76846 C46OFK 44343362 EC50 = 1.134 nM T76846 CL8Y3V 44343363 EC50 = 0.063 nM T76846 CCLF38 44347081 Ki = 5900 nM T76846 CT5V4X 44347082 Ki = 5900 nM T76846 C0QW9K 44347105 Ki = 1500 nM T76846 CWK01G 44347106 Ki = 3000 nM T76846 C4Y2SW 44347107 Ki = 20 nM T76846 C60PGA 44347110 Ki = 5900 nM T76846 CUEZ31 44347119 Ki = 56 nM T76846 CT03JB 44347219 Ki = 150 nM T76846 COD7W0 44347220 Ki = 29 nM T76846 CNP94O 44347221 Ki = 47 nM T76846 CBE37A 44347277 Ki = 420 nM T76846 CIZ30K 44347294 Ki = 190 nM T76846 C2YQM4 44347330 Ki = 5900 nM T76846 CX0Z1Y 44347331 Ki = 120 nM T76846 CAKI17 44347344 Ki = 0.23 nM T76846 CEIM86 44347370 Ki = 2.6 nM T76846 CS5ID0 44347378 Ki = 2900 nM T76846 CDN35X 44347379 Ki = 3000 nM T76846 CENG52 44347433 Ki = 14 nM T76846 CW1JY7 44347434 Ki = 0.96 nM T76846 C24GLU 44347435 Ki = 29 nM T76846 C7U2KM 44347838 IC50 = 3 nM T76846 CK6FH3 44347927 EC50 = 401 nM T76846 C58SIF 44348144 IC50 = 2900 nM T76846 C0F1EA 44348183 IC50 = 31 nM T76846 CC41MG 44348199 EC50 > 10000 nM T76846 CRSW34 44348200 EC50 = 2.8 nM T76846 C6E7SA 44349019 EC50 > 3000 nM T76846 C39SAR 44349173 IC50 = 2900 nM T76846 CZ4M3J 44349222 IC50 > 3500 nM T76846 CW9A4F 44349223 IC50 > 10000 nM T76846 C7RMI0 44349224 IC50 > 10000 nM T76846 CDW65K 44349226 IC50 > 8000 nM T76846 C3K9VR 44349228 IC50 > 10000 nM T76846 C7OW3R 44349246 IC50 > 10000 nM T76846 C26WVI 44349469 IC50 > 10000 nM T76846 CNB8U7 44349594 IC50 > 10000 nM T76846 C2QW1I 44364160 EC50 = 3.7 nM T76846 CLMA12 44366081 IC50 = 0.21 nM T76846 C2DHN5 44366155 IC50 = 110 nM T76846 CYD6R3 44366171 IC50 = 150 nM T76846 CO7U1L 44366182 IC50 = 41 nM T76846 CL4CY1 44366187 IC50 = 2.5 nM T76846 C9JN3L 44366213 IC50 = 190 nM T76846 C36FMV 44366215 IC50 = 0.19 nM T76846 CS27ZR 44366381 IC50 = 2.5 nM T76846 CQCP89 44387680 EC50 = 0.33 nM T76846 CD8HL0 44392514 Ki = 6500 nM T76846 CE21OM 44392535 Ki = 8800 nM T76846 C3IHV4 44393417 Ki = 5200 nM T76846 C2J1ML 44393418 Ki = 5600 nM T76846 CQ3L0D 44393421 Ki = 6800 nM T76846 C9C7SD 44393430 Ki = 114000 nM T76846 C47HVD 44393441 Ki = 15000 nM T76846 C1OG5U 44393450 Ki = 35000 nM T76846 CK5D8I 44394079 Ki = 2300 nM T76846 C25TVF 44394093 EC50 = 1340 nM T76846 C5K7CG 44394580 EC50 = 497 nM T76846 C08QML 44394581 EC50 = 473 nM T76846 C0OMU3 44394582 EC50 = 460 nM T76846 CL3P2Q 44394583 EC50 = 145 nM T76846 C5SGR6 44394584 EC50 = 886 nM T76846 CLXA10 44394585 EC50 = 863 nM T76846 C48NFW 44394586 EC50 = 961 nM T76846 C8GUD1 44394622 EC50 = 170 nM T76846 C9O4GM 44394623 EC50 = 4.7 nM T76846 C29ELZ 44394624 EC50 = 3 nM T76846 CP4A0B 44394625 EC50 = 553 nM T76846 C94PGA 44394626 EC50 = 2364 nM T76846 CF4O9U 44394627 EC50 = 827 nM T76846 CZ37TO 44394654 EC50 = 1016 nM T76846 CPE65R 44394655 EC50 = 3083 nM T76846 C9LKB5 44394656 EC50 = 1481 nM T76846 CG1Q8L 44394657 EC50 = 1449 nM T76846 CHG12Y 44394658 EC50 = 164 nM T76846 C9OTX4 44394659 EC50 = 3044 nM T76846 CNHD57 44394660 EC50 = 1013 nM T76846 CHTM92 44394689 EC50 = 913 nM T76846 C04RCL 44394690 EC50 = 452 nM T76846 CT9D5Y 44394691 EC50 = 313 nM T76846 CHDB95 44394692 EC50 = 992 nM T76846 CHZF38 44394693 EC50 = 43 nM T76846 C9Y6ZI 44394694 EC50 = 170 nM T76846 C06PXF 44394695 EC50 = 207 nM T76846 CJ97VD 44394730 EC50 = 757 nM T76846 C1IE7P 44394731 EC50 = 86.5 nM T76846 CLF0X5 44394732 EC50 = 175 nM T76846 C9QR1L 44394733 EC50 = 45 nM T76846 CP1IR5 44394734 EC50 = 556 nM T76846 C2UY8G 44394735 EC50 = 644 nM T76846 CTY36S 44394736 EC50 = 674 nM T76846 CR5B6L 44394748 EC50 = 1666 nM T76846 CW13LR 44394749 EC50 = 2635 nM T76846 CL3A0O 44394750 EC50 = 1604 nM T76846 CIGZ40 44394783 EC50 = 34.5 nM T76846 C62FUR 44394784 EC50 = 41 nM T76846 CCZ37I 44394785 EC50 = 203 nM T76846 C8RHG3 44394786 EC50 = 140 nM T76846 CQD01R 44394787 EC50 = 859 nM T76846 CO43JY 44394788 EC50 = 92.5 nM T76846 CCE30Z 44394789 EC50 = 6700 nM T76846 CVUQ61 44395681 Ki = 1400 nM T76846 CLT7X4 44396002 Ki = 1800 nM T76846 C8D2RU 44396986 IC50 = 2060 nM T76846 C6Z9BD 44396987 IC50 = 620 nM T76846 CZ2C9L 44397028 Ki = 650 nM T76846 CDZ3O4 44397030 Ki = 1100 nM T76846 C9V2RU 44397198 Ki = 710 nM T76846 C9CF7N 44397220 IC50 = 410 nM T76846 CXQ0M6 44397281 Ki = 3200 nM T76846 CPM68W 44397283 Ki = 2300 nM T76846 CX07ID 44397304 Ki = 2400 nM T76846 C7TNB6 44397410 IC50 = 940 nM T76846 C6F0QR 44397455 IC50 = 48 nM T76846 C49FRZ 44397461 EC50 = 2400 nM T76846 CNZ32D 44398259 IC50 = 158.49 nM T76846 C2YWK3 44398340 EC50 = 7.943 nM T76846 CJ36UT 44400660 Ki = 570 nM T76846 COM2E6 44400661 Ki = 1600 nM T76846 C56OUG 44400662 Ki = 950 nM T76846 CO7NM3 44400777 Ki = 830 nM T76846 C0E3XG 44400778 Ki = 810 nM T76846 C0OC7A 44400809 Ki = 860 nM T76846 COJM70 44400810 Ki = 450 nM T76846 CFT4O6 44400811 Ki = 1000 nM T76846 CC8SI2 44400813 Ki = 390 nM T76846 C3I0DM 44400814 Ki = 580 nM T76846 CAR95M 44400863 Ki = 1300 nM T76846 C2VI7C 44400864 Ki = 790 nM T76846 C2MEL4 44400932 Ki = 800 nM T76846 C61RQJ 44400934 Ki = 560 nM T76846 C2IJZ5 44400935 Ki = 670 nM T76846 CKH54Y 44401285 Ki = 900 nM T76846 C1JK9O 44401341 Ki = 10733 nM T76846 CTOS16 44401367 Ki = 66 nM T76846 CH1OX7 44401386 Ki = 2422 nM T76846 CR8GT9 44401392 Ki = 4861 nM T76846 CBQ7N3 44401418 Ki = 1486 nM T76846 CJNH94 44401440 Ki = 250 nM T76846 CUZJ52 44401513 Ki = 270 nM T76846 C9Y0LO 44401553 Ki = 871 nM T76846 C7E3YU 44401573 Ki = 1360 nM T76846 C5LID4 44401581 Ki = 692 nM T76846 CGNC86 44401587 Ki = 7061 nM T76846 C74QHS 44401592 Ki = 1110 nM T76846 CX30HI 44401607 Ki = 527 nM T76846 CRMV98 44408154 EC50 = 450 nM T76846 CIWX60 44408155 EC50 = 590 nM T76846 COG72Y 44408173 IC50 = 310 nM T76846 C3CQ4J 44408189 EC50 = 1200 nM T76846 CW08ZJ 44408190 IC50 = 460 nM T76846 CNWJ27 44408252 IC50 = 520 nM T76846 CH68SP 44408253 EC50 = 550 nM T76846 CCFV91 44408275 EC50 = 640 nM T76846 CZ3YG9 44408276 EC50 = 990 nM T76846 CAFP51 44408286 IC50 = 230 nM T76846 CR8HZ7 44408287 EC50 = 370 nM T76846 COC7D2 44408388 IC50 = 400 nM T76846 CJ4N3I 44409103 Ki = 23 nM T76846 C2NJ0V 44409104 Ki = 468 nM T76846 CKF52N 44409140 Ki = 2411 nM T76846 C5XEI8 44409206 Ki = 382 nM T76846 C9EXZ2 44409337 Ki = 24689 nM T76846 CFT41O 44409338 Ki = 6198 nM T76846 CUB1Q2 44409339 Ki = 55474 nM T76846 CK5GO1 44409379 Ki = 18016 nM T76846 C48WZD 44410802 Ki = 4600 nM T76846 C43IKV 44410803 Ki = 4200 nM T76846 C24AUD 44413828 EC50 = 214 nM T76846 C08PBM 44413829 EC50 = 286 nM T76846 CT4FW5 44413830 EC50 = 10 nM T76846 C8IDV1 44413831 EC50 = 3152 nM T76846 CZ3Q4T 44413832 Ki = 7163 nM T76846 CV6Z8C 44413842 EC50 = 2986 nM T76846 C4P0LS 44413879 EC50 = 340 nM T76846 C84OJQ 44413880 EC50 = 266 nM T76846 CN7I2S 44413881 Ki = 501 nM T76846 CF6O4K 44413913 EC50 = 563 nM T76846 CS42BM 44413914 EC50 = 15 nM T76846 CN18BL 44413930 Ki = 42 nM T76846 C4BMF6 44413931 EC50 = 42 nM T76846 C9WNH8 44413932 Ki = 219 nM T76846 CKZ86P 44413938 Ki = 154 nM T76846 CL2RK9 44413968 EC50 = 1474 nM T76846 CM2J9Z 44413969 Ki = 7441 nM T76846 C34XGB 44413970 Ki = 15358 nM T76846 C7IYH9 44415417 Ki = 1400 nM T76846 C3KQ8H 44415912 EC50 = 37 nM T76846 CDN97X 44415913 EC50 = 0.4 nM T76846 CAL83K 44415914 Ki = 1 nM T76846 C5CF0M 44415918 EC50 = 6 nM T76846 CXI18W 44415919 Ki = 1.1 nM T76846 C6DH7I 44415920 EC50 = 5.6 nM T76846 C06CYU 44415956 EC50 = 20000 nM T76846 CD2A9T 44415972 Ki = 1143 nM T76846 CHT4E8 44415991 Ki = 4122 nM T76846 CPX62S 44416014 Ki = 6107 nM T76846 C69CUX 44416057 EC50 = 0.5 nM T76846 C56DHI 44416060 EC50 = 163 nM T76846 CB2TU4 44416106 Ki = 7 nM T76846 CP9T4B 44416122 Ki = 461 nM T76846 C9KLB0 44416135 EC50 = 84 nM T76846 C37XPA 44416152 EC50 = 142 nM T76846 C1F7CU 44417402 IC50 > 1000 nM T76846 CBCR82 44417551 IC50 > 1000 nM T76846 CK0P4I 44417552 IC50 > 1000 nM T76846 CD72MS 44417553 IC50 > 1000 nM T76846 CT58RV 44417554 IC50 > 1000 nM T76846 C32QEO 44418413 EC50 > 10000 nM T76846 C7FEU6 44418420 EC50 > 10000 nM T76846 CZW07E 44418421 IC50 = 1.2 nM T76846 CLQG83 44418430 IC50 = 350 nM T76846 C8VG1S 44418431 IC50 = 5 nM T76846 C3HPI5 44418437 EC50 > 10000 nM T76846 CMD5N2 44418438 EC50 > 10000 nM T76846 CQE30X 44422937 IC50 = 860 nM T76846 C14FZP 44422938 IC50 > 2000 nM T76846 CE0H3Y 44422957 IC50 > 10000 nM T76846 C6H0NU 44422958 IC50 > 10000 nM T76846 C7I0KW 44422959 IC50 > 10000 nM T76846 C46XOB 44422960 IC50 > 10000 nM T76846 CNM90E 44422961 IC50 > 10000 nM T76846 C2K3BL 44422962 IC50 > 10000 nM T76846 C3E6VO 44422994 IC50 > 2000 nM T76846 CHU7G0 44422996 IC50 > 5000 nM T76846 C2LQW9 44422997 EC50 > 5000 nM T76846 CJM09S 44422998 IC50 > 5000 nM T76846 CI9HF1 44422999 EC50 = 1400 nM T76846 CXH5F8 44423009 IC50 = 990 nM T76846 C3VOD0 44423010 IC50 > 10000 nM T76846 C7UI3W 44423011 IC50 > 5000 nM T76846 CI05BD 44423012 IC50 > 10000 nM T76846 C5EJ3P 44423013 IC50 > 10000 nM T76846 C2NR7G 44423014 IC50 > 10000 nM T76846 CV3TL5 44423015 EC50 > 2500 nM T76846 CN5RD6 44431510 EC50 > 10000 nM T76846 CF3H8A 44431511 IC50 = 50 nM T76846 CVB07O 44431512 IC50 = 29 nM T76846 CY80GN 44431513 IC50 = 43 nM T76846 COCE51 44431515 EC50 = 1.85 nM T76846 CV62SP 44432932 Ki = 130 nM T76846 CL3ZR1 44432964 Ki = 4500 nM T76846 C0L4NV 44432966 Ki = 540 nM T76846 CKX7P2 44433264 Ki = 640 nM T76846 CZU4D1 44433294 Ki = 1100 nM T76846 CW8B6E 44433439 Ki = 1400 nM T76846 C8Z1IM 44434561 Ki = 289000 nM T76846 C5C6IA 44434562 Ki = 450 nM T76846 C6KPV5 44434568 Ki = 950 nM T76846 C2K9TI 44434570 Ki = 51000 nM T76846 CKL0H4 44434572 Ki = 65000 nM T76846 CKI3L6 44434580 Ki = 49000 nM T76846 CBC27H 44434581 Ki = 2700 nM T76846 C51NSB 44434584 Ki = 2100 nM T76846 CF2S6P 44434587 Ki = 1700 nM T76846 CQ81UI 44434592 Ki = 26000 nM T76846 CP2A4G 44434595 Ki = 104000 nM T76846 CT20IC 44434597 Ki = 30000 nM T76846 CC1H3U 44434598 Ki = 5700 nM T76846 CH17AO 44434599 Ki = 172000 nM T76846 CAID38 44434600 Ki = 65000 nM T76846 CGN1P8 44434601 Ki = 33000 nM T76846 CDV61Y 44434603 Ki = 18000 nM T76846 CZPC57 44434605 Ki = 63000 nM T76846 C5DT7Q 44434611 Ki = 48000 nM T76846 C3MS2D 44434613 Ki = 542000 nM T76846 C5A1GF 44434614 Ki = 45000 nM T76846 CN4D2E 44434616 Ki = 38000 nM T76846 C1B5RV 44434621 Ki = 19000 nM T76846 C5TMA6 44434625 Ki = 112000 nM T76846 C9XG2K 44434631 Ki = 106000 nM T76846 CY2C7G 44434632 Ki = 67000 nM T76846 CQ94YK 44434633 Ki = 32000 nM T76846 CM1NA8 44434634 Ki = 30000 nM T76846 C93NCL 44434635 Ki = 38000 nM T76846 CZ8TO1 44434636 Ki = 16000 nM T76846 CQ06DV 44434637 Ki = 47000 nM T76846 C3T4JG 44434639 Ki = 61000 nM T76846 C0SM2J 44434647 Ki = 25000 nM T76846 C9GIF5 44434648 Ki = 13000 nM T76846 CTQ16K 44434649 Ki = 5400 nM T76846 C15MAF 44434650 Ki = 27000 nM T76846 CWD27I 44434651 Ki = 27000 nM T76846 C6X8WB 44434652 Ki = 36000 nM T76846 CWU74N 44434653 Ki = 5400 nM T76846 CXN0M3 44434654 Ki = 27000 nM T76846 CM0VZ8 44434655 Ki = 22000 nM T76846 CV5Y3N 44434657 Ki = 41000 nM T76846 CVC93Q 44434658 Ki = 39000 nM T76846 CWE1V4 44434659 Ki = 162000 nM T76846 C5WR3A 44434661 Ki = 18000 nM T76846 CJ27QL 44434662 Ki = 15000 nM T76846 C6US7A 44434663 Ki = 47000 nM T76846 C4ZD1B 44434664 Ki = 106000 nM T76846 C03NKU 44434665 Ki = 43000 nM T76846 CJ2AT0 44434666 Ki = 3700 nM T76846 CF41SX 44434682 Ki = 26000 nM T76846 C9IWD4 44434683 Ki = 27000 nM T76846 CJ03PB 44434684 Ki = 43000 nM T76846 CIH0Z6 44434685 Ki = 36000 nM T76846 C4POB8 44434686 Ki = 46000 nM T76846 C1GFE6 44434687 Ki = 42000 nM T76846 C3J7WI 44434688 Ki = 28000 nM T76846 C9Y0BM 44434689 Ki = 24000 nM T76846 CH6LA5 44434690 Ki = 7100 nM T76846 CPRE40 44434691 Ki = 22000 nM T76846 C9O8LX 44434692 Ki = 23000 nM T76846 CE2Z3V 44434693 Ki = 16000 nM T76846 C31LUY 44434694 Ki = 26000 nM T76846 C9C4BN 44434695 Ki = 20000 nM T76846 CF3JX5 44434696 Ki = 55000 nM T76846 CM51SC 44434697 Ki = 14000 nM T76846 CA2FQ4 44434698 Ki = 46000 nM T76846 CTC18P 44434699 Ki = 249000 nM T76846 CQT85W 44434700 Ki = 201000 nM T76846 C8BQ7C 44434701 Ki = 22000 nM T76846 CV2QW3 44434702 Ki = 78000 nM T76846 C9IY3A 44434703 Ki = 121000 nM T76846 CF8J2P 44434704 Ki = 349000 nM T76846 CH7QD5 44434706 Ki = 220000 nM T76846 CT4FO2 44434707 Ki = 147000 nM T76846 C9E4PO 44434709 Ki = 80000 nM T76846 C7LUV2 44434713 Ki = 17000 nM T76846 CR70OD 44434714 Ki = 39000 nM T76846 CA1BF3 44434715 Ki = 9300 nM T76846 C0N4CY 44434753 Ki = 132000 nM T76846 CS1KG4 44434754 Ki = 37000 nM T76846 C2JHP0 44434757 Ki = 14000 nM T76846 CZ43DV 44434758 Ki = 94000 nM T76846 C50PIJ 44434759 Ki = 28000 nM T76846 CKAQ59 44434760 Ki = 22000 nM T76846 CALF38 44434761 Ki = 26000 nM T76846 C17HCY 44434762 Ki = 24000 nM T76846 CX75CS 44434763 Ki = 8300 nM T76846 CNB68V 44434764 Ki = 24000 nM T76846 CZ0R9M 44434765 Ki = 23000 nM T76846 CU9C0K 44434766 Ki = 12000 nM T76846 C8IHB1 44434767 Ki = 25000 nM T76846 C27KYV 44434768 Ki = 25000 nM T76846 CEM27N 44434769 Ki = 27000 nM T76846 CB7A2G 44434770 Ki = 52000 nM T76846 C0Y3IG 44434771 Ki = 65000 nM T76846 CNL2T3 44434772 Ki = 19000 nM T76846 CUW4Y6 44434778 Ki = 22000 nM T76846 CH8WT0 44434780 Ki = 278000 nM T76846 CL9K2D 44434781 Ki = 9400 nM T76846 CJ12GC 44434782 Ki = 16000 nM T76846 CFBX46 44434785 Ki = 8100 nM T76846 C0KB8P 44434787 Ki = 5400 nM T76846 C0M2VI 44434790 Ki = 57000 nM T76846 CH3UV8 44434794 Ki = 65000 nM T76846 C10VDG 44434797 Ki = 204000 nM T76846 CWN02S 44434799 Ki = 228000 nM T76846 C0X1MK 44434821 Ki = 7500 nM T76846 CU1ON8 44434828 Ki = 137000 nM T76846 CBHU73 44434839 Ki = 50000 nM T76846 C20UIF 44434841 Ki = 134000 nM T76846 CA7P5L 44434843 Ki = 9600 nM T76846 CBL2D7 44434845 Ki = 19000 nM T76846 CYE25C 44434847 Ki = 23000 nM T76846 CWE0J6 44434848 Ki = 17000 nM T76846 CB39YP 44434849 Ki = 45000 nM T76846 C0ZV6S 44434850 Ki = 40000 nM T76846 C4U6LJ 44434851 Ki = 44000 nM T76846 CA4M3C 44434853 Ki = 62000 nM T76846 CVGW87 44434854 Ki = 13000 nM T76846 C3G5QO 44434855 Ki = 4300 nM T76846 C2JET5 44434856 Ki = 78000 nM T76846 C2M5VB 44434857 Ki = 52000 nM T76846 CS30KD 44434858 Ki = 99000 nM T76846 C7S1OK 44434859 Ki = 31000 nM T76846 C3AVB5 44434860 Ki = 10000 nM T76846 CZQI93 44434861 Ki = 50000 nM T76846 CC0U5Y 44434862 Ki = 33000 nM T76846 CWTI58 44434863 Ki = 27000 nM T76846 CFOM13 44434864 Ki = 59000 nM T76846 CL97ID 44434865 Ki = 45000 nM T76846 CW93VX 44434867 Ki = 57000 nM T76846 CN36OD 44434868 Ki = 25000 nM T76846 CI09FJ 44434870 Ki = 29000 nM T76846 CZE48F 44434872 Ki = 30000 nM T76846 CXTV37 44434880 Ki = 25000 nM T76846 CQ45JU 44434884 Ki = 24000 nM T76846 CZ8H3M 44435220 Ki = 12000 nM T76846 C5D6YN 44441641 EC50 = 115 nM T76846 CP4TW0 44441642 EC50 = 680 nM T76846 CU6ZN4 44441644 EC50 = 263 nM T76846 CNS4O1 44441645 EC50 = 1001 nM T76846 CRL83D 44441646 EC50 = 840 nM T76846 C7EQ6Z 44441647 EC50 = 434 nM T76846 CHSV38 44441648 EC50 = 2950 nM T76846 CT3J4B 44441684 EC50 = 230 nM T76846 C3YRT9 44441685 EC50 = 241 nM T76846 CO93SX 44443035 Ki = 760 nM T76846 C1L7FO 44445109 Ki = 5.9 nM T76846 C08BMY 44448479 IC50 = 12240 nM T76846 C0C7KI 44448590 EC50 = 156.7 nM T76846 CQHR95 44448629 EC50 = 97.4 nM T76846 C78XDT 44448631 EC50 = 917.5 nM T76846 C8H1UT 44448660 EC50 = 249.9 nM T76846 CYAN15 44449216 IC50 = 1492 nM T76846 CTP3D6 44453826 Ki > 100000 nM T76846 C4FV3C 44453850 EC50 > 25000 nM T76846 CEI35V 44453902 Ki = 9100 nM T76846 CUPG04 44453903 Ki = 4500 nM T76846 C63APB 44456219 Ki = 1300 nM T76846 CE0P7K 44456222 Ki = 260 nM T76846 C5CIX6 44562287 Ki = 3100 nM T76846 CU92FG 44562414 Ki = 2300 nM T76846 CPSC21 44562440 Ki = 2500 nM T76846 CQ0I1K 44562460 Ki = 3100 nM T76846 CQ8J9K 44569175 EC50 = 25 nM T76846 CL8GU3 44569176 EC50 = 44 nM T76846 CD3T1I 44577060 Ki = 490 nM T76846 C6FI8E 44577062 Ki = 200 nM T76846 CJ6GZ3 44577063 Ki = 380 nM T76846 CWOK70 44577090 Ki = 570 nM T76846 C4FSH3 44577091 Ki = 190 nM T76846 CF8PL1 44577092 Ki = 160 nM T76846 CM6X5S 44577093 Ki = 220 nM T76846 CGTV08 44577094 Ki = 450 nM T76846 CEJ96P 44577510 EC50 = 2 nM T76846 CRSQ61 44577514 IC50 = 190 nM T76846 C6Y1BS 44577515 EC50 = 50 nM T76846 CM47HW 44577516 EC50 = 150 nM T76846 CHZ7Y6 44577518 IC50 > 10000 nM T76846 C5ZT9D 44577519 EC50 = 330 nM T76846 C8B1WR 44577520 EC50 = 56 nM T76846 CWFB17 44583567 EC50 = 2 nM T76846 CJB6H0 46203215 EC50 > 19100 nM T76846 CD3E4C 46885323 EC50 > 25200 nM T76846 CNW43Y 46885367 EC50 > 33300 nM T76846 CE4SF8 46885368 EC50 > 5720 nM T76846 CV23JL 46885415 EC50 = 500 nM T76846 CHPS01 46885417 EC50 > 14500 nM T76846 C4SVE1 46885480 EC50 = 71 nM T76846 C5QI7J 46885481 EC50 = 65 nM T76846 COU5X2 46885482 EC50 = 490 nM T76846 CG9NJ1 46885523 EC50 = 3660 nM T76846 CS90MN 46885524 EC50 = 7480 nM T76846 CQ94VM 46885526 EC50 = 4130 nM T76846 C90ABZ 46885558 EC50 = 600 nM T76846 C0MI3C 46885560 EC50 > 26700 nM T76846 C0Y9NF 46885711 EC50 = 3680 nM T76846 C3O5BR 46885712 EC50 = 3050 nM T76846 CG6XN0 46885759 EC50 = 570 nM T76846 CK8D6G 46885760 EC50 = 4570 nM T76846 C0C8GN 46885761 EC50 = 10700 nM T76846 CY30PG 46885815 EC50 > 33300 nM T76846 CEA70O 46885816 EC50 > 24700 nM T76846 CWN89S 46885863 EC50 > 33400 nM T76846 C8UTI7 46885907 EC50 > 13500 nM T76846 CFC5L1 46885972 EC50 = 11600 nM T76846 CO3S1Q 46905544 Ki = 7780 nM T76846 C96XEU 46905545 Ki = 11250 nM T76846 C29LQB 46919520 IC50 = 482.7 nM T76846 C1EMQ2 49861348 EC50 = 1160 nM T76846 C9QU3G 49862375 EC50 = 90 nM T76846 CPZI97 49862377 EC50 = 79 nM T76846 CY7R2T 49862378 EC50 = 880 nM T76846 C7GA4I 49862425 EC50 = 2500 nM T76846 C0QD9I 51346770 Ki = 1182 nM T76846 C30PGL 51346771 Ki = 4530 nM T76846 CBQN64 52918026 IC50 = 650 nM T76846 CG5TJ0 53240339 IC50 = 400 nM T76846 C6GET3 54582029 IC50 = 500 nM T76846 CQ7O3U 54584301 IC50 = 760 nM T76846 C8PIL3 54584302 IC50 = 740 nM T76846 CN6F2C 54586246 IC50 = 390 nM T76846 CEU0M6 54587278 IC50 = 33 nM T76846 C2WAO4 57634921 Ki = 45 nM T76846 C4VT5C 57634925 Ki = 22 nM T76846 CKW2T0 57646411 Ki = 2 nM T76846 C8F5XG 57646441 Ki = 2.5 nM T76846 CH1LU3 58777892 Ki = 8200 nM T76846 CS27GN 70682904 Ki = 104000 nM T76846 C73SKU 70682946 IC50 = 25 nM T76846 CPJ08L 70688853 Ki = 8 nM T76846 C2O7TA 71449047 IC50 = 130 nM T76846 CH0F4A 71449048 IC50 = 5600 nM T76846 CMS5R6 71449140 Ki = 752000 nM T76846 CKCN10 71452720 IC50 = 620 nM T76846 CEB0P9 71452732 Ki = 1200 nM T76846 CY16AM 71454518 Ki = 19000 nM T76846 CPX03G 71456219 IC50 = 200 nM T76846 C07WXP 71456220 IC50 = 620 nM T76846 CNRV69 71456245 IC50 = 1600 nM T76846 CU17GR 71458055 Ki = 500 nM T76846 C6YR0U 71458117 IC50 > 10000 nM T76846 CJ52CU 71459938 EC50 = 1100 nM T76846 CU2A1J 71461601 EC50 = 98 nM T76846 CECQ16 71461657 Ki = 1200 nM T76846 C24GWM 71461662 Ki = 52000 nM T76846 CZ94CM 71461730 EC50 = 27.6 nM T76846 CYA8G1 71717886 EC50 = 13 nM T76846 CV8K5U 73345513 Ki = 3400 nM T76846 C4IAM6 73345514 Ki = 12 nM T76846 C1A5SK 73345616 IC50 > 10000 nM T76846 CI0DV9 73345617 IC50 > 5000 nM T76846 CD1NE3 73345618 EC50 > 500 nM T76846 CYMH60 73347015 Ki = 25 nM T76846 CZ91TE 73347138 EC50 = 370 nM T76846 CK46SP 73347139 IC50 = 4400 nM T76846 CX9LF8 73347140 IC50 > 1000 nM T76846 C4SR8Z 73348617 EC50 = 11 nM T76846 CS4I5R 73350057 Ki = 1.2 nM T76846 CMLR03 73350220 IC50 = 270 nM T76846 C3EF0P 73351617 Ki = 0.2 nM T76846 CKWH98 73351727 IC50 = 3900 nM T76846 C1L7HK 73353100 Ki = 0.81 nM T76846 CJL0D3 73353101 EC50 = 150 nM T76846 C8C0LW 73353205 IC50 > 10000 nM T76846 CGVC68 73353206 IC50 > 1000 nM T76846 CK2X0G 73353271 IC50 = 290 nM T76846 CK23FW 73354573 Ki = 20 nM T76846 CIEJ89 73354618 Ki = 15 nM T76846 C0ISQ4 73354708 IC50 = 630 nM T76846 CJS25D 73354709 IC50 > 10000 nM T76846 C7OT4D 73354780 EC50 = 5.4 nM T76846 C17PEL 73356313 IC50 = 6.7 nM T76846 CR7OX0 90664763 EC50 = 2900 nM T76846 C6L8AD 101043841 IC50 = 590 nM T76846 C1KS2F 101043843 EC50 = 1.9 nM T76846 CI8PR4 118718122 EC50 = 2 nM T76846 CCL46X 118718855 IC50 > 10000 nM T76846 CK6FL5 118718881 EC50 = 161.4 nM T76846 C8ME0B 118735099 EC50 = 52 nM T76846 CK17XF 118735100 IC50 = 5000 nM T76846 C1O7GU 118735101 IC50 = 100 nM T76846 CBTC79 118735102 EC50 = 2000 nM T76846 C1O3GL 118735103 EC50 = 55 nM T76846 C65WMB 122184498 IC50 = 3.74 nM T76846 CH9L8O 122184499 IC50 = 23 nM T76846 CAQ17N 122184571 IC50 = 20.4 nM T76846 CK48WX 122184572 IC50 = 47.4 nM T76846 CF9PO7 122184573 IC50 = 27.4 nM T76846 C3FBZ9 122184574 IC50 = 3.2 nM T76846 CCP0X7 122184575 IC50 = 17.8 nM T76846 C7OBX1 122184576 IC50 = 1.6 nM T76846 CU73AF 122184577 EC50 = 709 nM T76846 CGB7F4 122184578 IC50 = 24.9 nM T76846 CB7HZ8 122184579 EC50 = 463 nM T76846 C9HE4L 122184580 EC50 = 9.92 nM T76846 C9MJT7 122184581 EC50 = 16 nM T76846 C20NAY 122184582 EC50 = 13.2 nM T76846 CH1B8W 122184631 IC50 = 15.3 nM T76846 CLXB63 122184632 IC50 = 547 nM T76846 CIJ14O 122184633 IC50 = 9.7 nM T76846 CDSR31 122184634 IC50 = 147 nM T76846 CL28BX 122184635 EC50 = 11 nM T76846 CYOR02 122184636 IC50 = 8 nM T76846 C09LFS 122184637 IC50 = 2.5 nM T76846 C5CDX9 122184638 EC50 = 1790 nM T76846 C64BPZ 122184639 EC50 = 1.47 nM T76846 CEDT39 122184640 EC50 = 802 nM T76846 CLB43S 122184641 EC50 = 753 nM T76846 CN4L5U 122184908 IC50 = 336 nM T76846 CG0U7B 122184909 IC50 = 1270 nM T76846 CZ4HW7 122184910 EC50 = 326 nM T76846 C6KW7J 122184911 EC50 = 5180 nM T76846 CK3VM5 122184912 EC50 = 770 nM T76846 C0AFH9 122184913 IC50 = 657 nM T76846 CNBA05 122184914 EC50 = 1400 nM T76846 C7CLU6 133053557 EC50 = 30 nM T76846 CJNF06 137631599 EC50 = 204.17 nM T76846 COM8N7 137631628 IC50 = 17 nM T76846 CW9P1D 137633115 EC50 = 521 nM T76846 CF2NA9 137633806 EC50 = 30.9 nM T76846 CTD90C 137634090 EC50 = 22000 nM T76846 CPL59T 137635422 EC50 = 122.6 nM T76846 CM1H6A 137636428 EC50 > 3000 nM T76846 CU4KL7 137636677 EC50 = 8709.64 nM T76846 CVC3Q2 137636965 EC50 = 5370.32 nM T76846 CK2CZ3 137637026 EC50 = 160 nM T76846 CME01A 137637283 EC50 = 5.1 nM T76846 C6TKX9 137637656 EC50 = 633.1 nM T76846 CMJ4I7 137637705 IC50 = 117 nM T76846 C2FEA6 137638725 Ki > 1000 nM T76846 CH17TL 137638778 EC50 = 19.4 nM T76846 CZ74WU 137639140 EC50 > 100000 nM T76846 CKR14I 137639770 EC50 = 6.7 nM T76846 CHB9X0 137640703 EC50 = 6918.31 nM T76846 CBL5Z9 137641157 EC50 = 467.74 nM T76846 CCPD94 137641398 EC50 = 309.03 nM T76846 CTN96O 137642298 EC50 > 1000 nM T76846 CGP0V3 137643023 EC50 > 3000 nM T76846 CAT50J 137643076 IC50 > 1000 nM T76846 C5R2TI 137643266 IC50 = 56 nM T76846 CE0YF4 137643385 EC50 > 3000 nM T76846 C68AYB 137644225 EC50 > 3000 nM T76846 CJ1I7B 137645567 Ki > 100000 nM T76846 CT18GM 137646617 EC50 = 7413.1 nM T76846 CV5RX4 137647009 EC50 = 721.6 nM T76846 CY7K4J 137647538 EC50 = 758.58 nM T76846 C10VFY 137648144 EC50 = 821.3 nM T76846 C5X7AK 137648344 IC50 > 1000 nM T76846 CSF97J 137649543 EC50 > 3000 nM T76846 CIV6Z7 137649910 EC50 > 3000 nM T76846 C7I9CK 137651025 EC50 > 100000 nM T76846 CF3VP0 137651074 EC50 = 5 nM T76846 CH62TM 137653176 EC50 > 3000 nM T76846 CF5Z2W 137653739 EC50 = 0.8 nM T76846 CKX3Q9 137653925 EC50 = 26915.35 nM T76846 CMO01K 137655905 EC50 = 2137.96 nM T76846 CKL0Y8 137656033 EC50 > 3000 nM T76846 C5WHL4 137656521 EC50 = 290.6 nM T76846 CJ9RO7 137657609 IC50 = 18 nM T76846 C5FI6X 137657633 IC50 = 40 nM T76846 COS0A1 137658158 EC50 = 1479.11 nM T76846 CS1PR7 137659394 EC50 > 1000 nM T76846 CHB32J 137659790 EC50 = 2691.53 nM T76846 CQ7S0L 137659949 EC50 > 100000 nM T76846 C2XLI7 137660671 EC50 = 1000 nM T76846 C98FVD 137660993 EC50 = 20.42 nM T76846 C4CFP9 137661893 EC50 >= 1910 nM T76846 CCZ72V 137662147 EC50 = 161.7 nM T76846 C2WC5J 145948876 EC50 = 42 nM T76846 CUC3S2 145948912 IC50 = 580 nM T76846 C8D7OM 145964017 EC50 = 76 nM T76846 CCK75J 145964837 IC50 = 14 nM T76846 CS73TM 145966364 EC50 = 1 nM T76846 CHU51B 145966490 EC50 = 12 nM T76846 CJO1Y6 145966716 EC50 = 3.2 nM T76846 C9RA7Q 145967155 IC50 = 2.2 nM T76846 CICD84 145971389 EC50 = 1.8 nM T76846 C97DEG 145971673 EC50 = 276 nM T76846 CEV4F6 145972289 EC50 = 5 nM T76846 C9NRU8 145973779 IC50 = 4.4 nM T76846 CYD0J5 145973975 EC50 = 1.9 nM T76846 CR2NQ5 145975465 IC50 = 20 nM T76846 CKP26E 145976444 EC50 = 19 nM T76846 C7UJ8Q 145976863 EC50 = 4.1 nM T76846 CMS17N 145977650 IC50 = 11 nM T76846 CJ28PL 145980198 EC50 = 255 nM T76846 C0S1IN 145980719 EC50 = 120 nM T76846 CEZU78 145980838 IC50 > 1000 nM T76846 CM5UX9 145981147 IC50 > 1000 nM T76846 CJ5T1Y 145987870 IC50 = 46.8 nM T76846 CF34MX 145988152 EC50 = 57 nM T76846 C39KYZ 145988867 EC50 = 315 nM T76846 C7WF3R 145989222 EC50 = 116 nM T76846 C50ZLS 145990599 IC50 = 90 nM T76846 CRSZ36 145993132 EC50 > 1000 nM T76846 CDQZ25 145994283 EC50 > 1000 nM T76846 C10FUX 145994325 IC50 > 5000 nM T76846 C5S4PT 24858479 EC50 > 5000 nM T76846 CA83CB 24858481 EC50 > 4000 nM T76846 CR08PO 24858629 IC50 = 380 nM T76846 D00TSX 11672424 IC50 = 12 nM T76846 D00VYC 44400370 Ki = 55.02 nM T76846 D01HTX 11707715 IC50 = 250 nM T76846 D01VMU 44445082 EC50 = 29 nM T76846 D02JVA 44408515 IC50 = 2.6 nM T76846 D02MPZ 11535237 EC50 = 37 nM T76846 D03AZC 25078192 Ki = 1.44 nM T76846 D04BOG 11629290 EC50 > 10000 nM T76846 D04YZZ 44445083 IC50 = 11 nM T76846 D05LLI 11498895 IC50 = 1.4 nM T76846 D05WNC 11520823 IC50 = 140 nM T76846 D05XRI 44400401 EC50 = 0.68 nM T76846 D06PNU 44409257 Ki = 1632 nM T76846 D06RTP 11700730 IC50 = 1.7 nM T76846 D07DWH 44400402 EC50 = 1.61 nM T76846 D07IBF 44400322 Ki > 500 nM T76846 D07SFD 44408443 EC50 = 1.2 nM T76846 D07UXW 44408400 IC50 = 820 nM T76846 D08DND 44445084 IC50 = 84 nM T76846 D09OMI 44400400 Ki = 97.97 nM T76846 D09PDT 24774519 IC50 = 32 nM T76846 D09UUC 46877881 Ki = 390 nM T76846 D09XCH 44400371 Ki > 500 nM T76846 D0A8ME 44400398 Ki = 399.7 nM T76846 D0B8GR 44413876 EC50 = 541 nM T76846 D0B9NH 44408399 EC50 = 4300 nM T76846 D0C7VI 44400369 Ki = 7.91 nM T76846 D0F6GX 44409240 Ki = 1727 nM T76846 D0GN9K 24774602 EC50 = 27 nM T76846 D0L1MJ 11700739 IC50 = 6 nM T76846 D0M4EF 11593084 EC50 = 27 nM T76846 D0N6KO 9938402 Ki = 125 nM T76846 D0P4GI 11629326 IC50 = 13 nM T76846 D0QW4A 24774356 EC50 = 95 nM T76846 D0R0BY 44400320 Ki = 3.12 nM T76846 D0U5KM 11093672 EC50 = 7.1 nM T76846 D0VD7R 44408408 IC50 = 2700 nM T76846 D0W1SM 44408413 IC50 = 270 nM T76846 D0WG8P 44400321 Ki = 15.87 nM T76846 D0WI8M 44445085 IC50 = 12 nM T76846 D0X1YL 25078242 Ki = 166.41 nM T76846 D0XQ5U 24774438 IC50 = 23 nM T76846 D0YB7F 92432 EC50 = 0.2042 nM T76846 D0ZD3M 44400399 Ki = 313.48 nM T29999 D0F4NS 119369 IC50 = 2000 nM T29999 D02RDE 9939929 IC50 = 3 nM T29999 D08ORO 114904 IC50 = 440 nM T29999 C4V2XT 9939024 IC50 < 1 nM T29999 CM7Q1K 10578000 IC50 = 400 nM T29999 CFP17Y 10578460 IC50 = 700 nM T29999 CR01ZV 10603742 IC50 > 10000 nM T29999 CSP1C3 10626339 IC50 = 400 nM T29999 C58XOT 10840974 IC50 = 1000 nM T29999 C4C8QJ 11158261 IC50 = 4 nM T29999 CZWJ61 11167861 IC50 = 2000 nM T29999 C4JKH8 11190868 IC50 = 490 nM T29999 CB43VY 11239468 IC50 = 10 nM T29999 C9Q7RV 11262100 IC50 = 5 nM T29999 CE0DX4 11269308 IC50 = 4000 nM T29999 CZ0JW9 11270497 IC50 = 2100 nM T29999 C89CZT 11272841 IC50 = 800 nM T29999 CTP85J 11317662 IC50 = 50 nM T29999 CFU2E1 11351397 IC50 = 210 nM T29999 CN2YM9 11365307 IC50 = 2200 nM T29999 CON43W 11386922 IC50 = 3000 nM T29999 CHRT50 11397211 IC50 = 60 nM T29999 C93VQG 11418441 IC50 = 290 nM T29999 CPG63Z 11422294 IC50 = 50 nM T29999 CN14VO 11476070 IC50 = 2900 nM T29999 CIS2N6 11490514 IC50 = 5 nM T29999 CZ3PM4 11490613 IC50 = 10 nM T29999 COJ27D 11763684 IC50 = 50 nM T29999 CQ5SR1 15285180 IC50 = 600 nM T29999 CWRJ17 15285181 IC50 = 3300 nM T29999 C7D8XH 21467167 IC50 = 300 nM T29999 CJBV97 44386548 IC50 = 780 nM T29999 CP9TR0 10324985 Ki > 10000 nM T62206 C28QWT 17498 Ki = 30000 nM T62206 CX3EK0 1369939 IC50 = 500 nM T62206 CJH21V 20836008 Ki = 1000 nM T62206 C4J1KV 101873572 IC50 = 1500 nM T62206 CV0ES8 118709594 IC50 = 10000 nM T62206 C6FIT4 118885449 IC50 = 2800 nM T62206 C84WVJ 118885459 IC50 = 2300 nM T62206 CVX7S9 118885461 IC50 = 1100 nM T62206 CU2F8K 118885471 IC50 = 2300 nM T62206 C4VRT3 118886849 IC50 = 300 nM T62206 C8Q0ED 118886853 IC50 = 5600 nM T62206 C8LNZ4 118886858 IC50 = 250 nM T62206 C4C0MT 118886861 IC50 = 1400 nM T62206 CRQ48Z 118886862 IC50 = 900 nM T62206 CNW7P4 118886864 IC50 = 201.7 nM T62206 CZR09C 122198706 IC50 = 4800 nM T62206 C7J8VG 145969348 IC50 = 11200 nM T62206 C46VCD 145969980 IC50 = 8300 nM T62206 C4WL7R 145970220 IC50 = 1600 nM T62206 C4U2MG 155565853 EC50 = 6040 nM T62206 D0EJ9B 66827 Ki = 470000 nM T07217 D06RWL 58448012 IC50 = 6340 nM T07217 D08SNH 71555922 Ki = 7 nM T07217 CB3K6A 96214 IC50 = 4000 nM T07217 C46KNF 521274 IC50 = 16800 nM T07217 C4FC1N 626798 Ki = 105 nM T07217 CA6J5T 710279 IC50 = 4400 nM T07217 CVE5Y3 736244 IC50 > 100000 nM T07217 CF8D7G 803793 Ki > 1400 nM T07217 CW15QO 985472 IC50 > 100000 nM T07217 CGW4J2 1078969 IC50 > 100000 nM T07217 CRJ5C4 1201248 Ki = 2500 nM T07217 CMF16D 1309516 Ki = 2300 nM T07217 CL3B7X 2729589 IC50 > 100000 nM T07217 CP1O4I 2732293 IC50 = 1000 nM T07217 C4KHI2 2799758 IC50 > 100000 nM T07217 CHN96D 2808809 IC50 > 100000 nM T07217 CPV39W 2809956 IC50 > 100000 nM T07217 CI0X5C 2810912 IC50 > 100000 nM T07217 CP17LN 2811714 IC50 = 3100 nM T07217 CX4B0Q 2815870 IC50 > 100000 nM T07217 C3O1JG 2859016 Ki = 290 nM T07217 CH0Q2K 2869257 Ki = 380 nM T07217 CK4Y1N 3113729 Ki = 690 nM T07217 CIM4D6 3125032 Ki = 5400 nM T07217 C51ISE 4533882 Ki = 610 nM T07217 C5J2VI 9803569 Ki = 12 nM T07217 C8UM5T 9863791 IC50 = 69 nM T07217 CBE76H 9889814 Ki = 6 nM T07217 CD07HS 9908257 IC50 = 49 nM T07217 C1VF3H 9970420 IC50 = 430 nM T07217 C09XCF 9996070 IC50 = 96 nM T07217 C8HD1X 10001781 Ki = 58 nM T07217 CZ0G7C 10017976 IC50 = 590 nM T07217 CVT8H1 10019079 IC50 < 400 nM T07217 CUQI21 10022216 IC50 < 400 nM T07217 CJ4Y6Z 10031785 IC50 = 7900 nM T07217 CYU01B 10064783 IC50 = 830 nM T07217 CMZ32I 10065528 IC50 = 550 nM T07217 C0RP7J 10088310 IC50 = 2680 nM T07217 C3TF8H 10246342 IC50 = 600 nM T07217 C0T6KH 10248758 IC50 = 2390 nM T07217 CUN7D5 10384708 IC50 = 1660 nM T07217 CCV23K 10426344 IC50 < 400 nM T07217 CE58QI 10471204 IC50 = 1090 nM T07217 CUOL84 11722643 IC50 = 750 nM T07217 CN9I5J 12020821 Ki < 2 nM T07217 CO7Z8E 12020835 Ki = 3.4 nM T07217 C0G6VU 14576198 IC50 = 1100 nM T07217 C7EW5A 15944037 Ki = 1280 nM T07217 C9DR4J 15944049 Ki = 400 nM T07217 CTCI07 16773270 Ki = 4320 nM T07217 CQ81TK 17753148 Ki < 2 nM T07217 CGY78B 20105362 Ki = 4300 nM T07217 C06GWX 20577249 Ki < 2 nM T07217 CN7GB8 20577253 Ki > 2000 nM T07217 C1WJA3 20577258 Ki = 130 nM T07217 C7GJ4F 20577259 Ki = 2.7 nM T07217 C6R9WC 20577264 Ki = 3.5 nM T07217 C93VWY 20577272 Ki = 9.3 nM T07217 CUK06Z 20577273 Ki = 18 nM T07217 C5USN9 20577275 Ki = 36 nM T07217 C2HX1C 22258075 Ki = 50 nM T07217 C5N6GX 22258086 Ki < 2 nM T07217 CU3E1A 28828687 Ki = 4840 nM T07217 CRH19V 43084137 Ki = 6510 nM T07217 CK4G3W 43084211 Ki = 2550 nM T07217 C5PT0H 44393551 IC50 = 32000 nM T07217 CQ2YZ1 44393553 IC50 = 2600 nM T07217 CG8SX9 44393559 IC50 = 2600 nM T07217 C4MQV8 44393578 IC50 = 4500 nM T07217 C7PHW4 44393579 IC50 = 1300 nM T07217 CXB68V 44393608 IC50 = 3500 nM T07217 C01GWF 44393609 IC50 = 4700 nM T07217 C16FLV 44393613 IC50 = 30000 nM T07217 CZEL27 44393682 IC50 = 89000 nM T07217 CP1F0B 44393712 IC50 > 100000 nM T07217 CJFA96 44393738 IC50 = 10000 nM T07217 CU7RC3 44393763 IC50 = 7100 nM T07217 C5Z6CG 44393764 IC50 = 1300 nM T07217 CS5BL9 44393786 IC50 = 1500 nM T07217 C1W9HS 44393788 IC50 = 7400 nM T07217 CWAK75 44393806 IC50 = 13000 nM T07217 CGC3D4 44393811 IC50 = 1100 nM T07217 C61CQG 44414921 Ki > 2000 nM T07217 CM5P0D 44441313 Ki = 28 nM T07217 CV8QE2 44441314 Ki = 650 nM T07217 CHW12X 44564601 IC50 = 1810 nM T07217 CFA64Q 44564613 IC50 > 25000 nM T07217 C0WIG2 44564614 IC50 = 970 nM T07217 CJOY69 44564615 IC50 = 670 nM T07217 CAF14Y 44564616 IC50 = 710 nM T07217 CYJ21U 44564617 IC50 = 720 nM T07217 CAM24R 44564618 IC50 = 780 nM T07217 CI82XK 44564826 IC50 > 25000 nM T07217 C9CM8I 44564869 IC50 = 1040 nM T07217 C4E7MC 44564870 IC50 = 2030 nM T07217 CD8CT3 44564871 IC50 < 400 nM T07217 CTNH09 46890483 IC50 = 56300 nM T07217 CC82RP 49871914 Ki = 32 nM T07217 CCNW31 49871916 Ki = 7 nM T07217 CC91VI 49872007 Ki = 5 nM T07217 C47ASG 49872008 Ki < 1 nM T07217 C2UY0W 49872009 Ki = 6 nM T07217 COJ51Y 49872404 Ki < 1 nM T07217 CAJ79L 49872405 Ki = 13 nM T07217 CAJ6O2 62033065 Ki = 1190 nM T07217 CW6AX8 62034157 Ki = 1950 nM T07217 C7A8GR 62034326 Ki = 2690 nM T07217 C9P5KT 71556166 Ki = 12 nM T07217 C8JOU5 71556223 Ki = 22 nM T07217 C25XGY 71556353 Ki = 16 nM T07217 CP0J5L 71556425 Ki = 11 nM T07217 CB5QR3 71556493 Ki = 13 nM T07217 CIXL34 71556883 Ki = 20 nM T07217 CZ3A7E 71556887 Ki = 16 nM T07217 CH4SQ1 71567114 IC50 > 10000000 nM T07217 CQV78J 71567246 IC50 = 6130 nM T07217 CO5TP2 71567247 IC50 = 74000 nM T07217 C2R5DV 71567248 IC50 = 31000 nM T07217 CJ46DW 71567249 IC50 = 5410 nM T07217 CJ3IH9 71567250 IC50 = 9510 nM T07217 C89VKW 71567251 IC50 = 3020 nM T07217 CEXH43 71567376 IC50 = 6390 nM T07217 CHJ50Z 71567377 IC50 = 259000 nM T07217 CV2O3U 71567378 IC50 = 86000 nM T07217 CV6R9I 71567379 IC50 = 10200 nM T07217 CSH09F 71567380 IC50 = 5640 nM T07217 CZ4FD0 71567381 IC50 = 4320 nM T07217 CZQM42 71567505 IC50 = 10300 nM T07217 CMH1D4 71567506 IC50 = 13600 nM T07217 CZ95BC 71567507 IC50 = 4270 nM T07217 C1NMO8 71567509 IC50 = 2500 nM T07217 CTX12Q 71567510 IC50 = 16600 nM T07217 C8LI9S 71567642 IC50 = 23500 nM T07217 CGU46H 71567643 IC50 = 15500 nM T07217 C2I7UL 71746991 IC50 = 82800 nM T07217 CC53VS 71746992 IC50 = 14800 nM T07217 CD9J0Z 71746994 IC50 = 14800 nM T07217 COJ59Z 71746995 IC50 > 100000 nM T07217 CQ30LW 72695132 Ki = 120 nM T07217 CYC78V 72722031 Ki = 100 nM T07217 C67HRP 73553418 Ki = 350 nM T07217 C6ECV1 121225428 Ki = 30 nM T07217 CSHO57 127045592 Ki = 3100 nM T07217 CMZ3V8 134158371 Ki = 210 nM T07217 C5AKN4 134158372 Ki = 200 nM T07217 C4MX6V 134158373 Ki = 7750 nM T07217 CHRZ86 134158374 Ki = 590 nM T07217 CQG2S9 134158375 Ki = 1160 nM T07217 CI4QH1 135432878 IC50 = 2900 nM T07217 CW80LM 135440059 IC50 = 1000 nM T07217 C48XTV 135459601 IC50 > 100000 nM T07217 CZJ37D 135521816 Ki = 10300 nM T07217 CW0V5I 135587623 Ki = 3600 nM T07217 C46KFZ 135713542 IC50 = 47000 nM T07217 CNQX23 135727209 IC50 > 100000 nM T07217 C9BA7U 135815067 IC50 = 600 nM T07217 CLK5Q8 135816280 IC50 > 100000 nM T07217 CL0FM8 136048711 IC50 = 24000 nM T07217 CRP6A8 136048712 IC50 = 3900 nM T07217 CF80BT 136048713 IC50 = 33000 nM T07217 C3JCM4 136048714 IC50 > 100000 nM T07217 CTVD48 136048715 IC50 > 100000 nM T07217 CMOE09 136048716 IC50 = 33000 nM T07217 CCB5I9 136048717 IC50 = 4000 nM T07217 C2SUF4 136048718 IC50 = 23000 nM T07217 C8X7UL 136048719 IC50 = 33000 nM T07217 C06ZLA 136048720 IC50 = 25000 nM T07217 CF1O3N 136048721 IC50 = 37000 nM T07217 C2H7FU 136048722 IC50 > 100000 nM T07217 C5K4ND 136048723 IC50 > 100000 nM T07217 C58QAB 136048724 IC50 > 100000 nM T07217 CY05IB 145980493 Ki = 760 nM T07217 CA3KT7 145980569 Ki = 230 nM T07217 C1ASQ2 145980794 Ki = 910 nM T07217 C0Q8AN 145980978 Ki = 2120 nM T07217 C3PW5C 145981329 Ki > 6140 nM T07217 CASL30 145981654 Ki = 930 nM T07217 CDYB12 145982036 Ki = 580 nM T07217 C1GHW8 145984604 Ki = 1850 nM T07217 CBL2O5 145986398 Ki > 6140 nM T07217 CF5C8E 145986667 Ki > 6140 nM T07217 CSNM96 145987716 Ki = 1670 nM T07217 CK6LC5 145988577 Ki = 840 nM T07217 C2BP4Y 145988687 Ki > 6140 nM T07217 CD13VT 145989763 Ki > 6140 nM T07217 CS47GH 145991412 Ki = 2160 nM T07217 C62QNV 145992166 Ki = 820 nM T07217 CK7V8N 145992248 Ki = 1150 nM T07217 C1OC7T 145992458 Ki = 2760 nM T07217 CNPT68 145993480 Ki = 7380 nM T07217 CX9MH4 145994114 Ki > 6140 nM T07217 CR4SP9 155510891 IC50 = 1700 nM T07217 CW7Y8D 155511415 IC50 = 2980 nM T07217 CC7RL2 155517237 IC50 = 1890 nM T07217 C0W7OZ 155517587 IC50 = 1970 nM T07217 CR65JX 155520458 IC50 = 3590 nM T07217 C8PM9B 155524334 IC50 = 2300 nM T07217 C2ZVO6 155525963 IC50 = 2370 nM T07217 CS7IZ8 155526071 IC50 = 2430 nM T07217 C4KX9C 155528528 IC50 = 14780 nM T07217 CAT83B 155528650 IC50 = 1190 nM T07217 C7SEQ6 155530621 IC50 = 4040 nM T07217 CA90NS 155532366 IC50 = 2990 nM T07217 CDP93T 155532593 IC50 = 2640 nM T07217 C1I3BM 155535681 IC50 = 2200 nM T07217 C3CDA5 155539479 IC50 = 1580 nM T07217 C9BD0X 155546393 IC50 = 1740 nM T07217 CV3TE6 155549399 IC50 = 3530 nM T07217 C84GMX 155554918 IC50 = 4730 nM T07217 C7ITE5 155555180 IC50 = 4380 nM T07217 C1SCP4 155555555 IC50 = 24830 nM T07217 C2J5FB 155555976 IC50 = 3150 nM T07217 C8RX9K 155556798 IC50 = 1190 nM T07217 C8TO2H 155559803 IC50 = 3540 nM T07217 CTL1V7 155568705 IC50 = 2410 nM T07217 CW01DA 44441441 Ki = 2 nM T07217 D00ORM 28971834 IC50 = 800 nM T07217 D02TVS 985 Ki = 336 nM T07217 D03DUX 44393606 IC50 = 12000 nM T07217 D03LOG 5280450 IC50 = 1000 nM T07217 D05GVL 44393683 IC50 = 6100 nM T07217 D05JAH 448769 IC50 = 570 nM T07217 D06BBB 16122583 Ki < 2 nM T07217 D07OKT 219301 IC50 = 9400 nM T07217 D08KLL 10126984 Ki = 16 nM T07217 D0A4EA 445639 Ki = 185 nM T07217 D0B9SJ 5714537 Ki = 670 nM T07217 D0C1DG 44393734 IC50 = 4300 nM T07217 D0C7RS 1369 Ki = 1000 nM T07217 D0H2UM 44393643 IC50 = 12000 nM T07217 D0I1RP 44393638 IC50 = 10000 nM T07217 D0WF7I 16046219 Ki = 2.5 nM T07217 D0Y8JN 44393556 IC50 = 8500 nM T07217 D0YW9C 44564825 IC50 = 3600 nM T13259 D00BRD 126 IC50 = 24700 nM T13259 D09SWE 31244 IC50 > 1000000 nM T13259 D0B5YS 1183 IC50 = 15600 nM T13259 D0NH9P 135 IC50 > 1000000 nM T13259 D0X7BT 125 IC50 > 1000000 nM T13259 C6X9CB 978 IC50 > 1000000 nM T13259 C0F1EW 6271 IC50 = 293000 nM T13259 CV9N2M 7469 IC50 = 166000 nM T13259 CR0U3Y 115067 IC50 > 1000000 nM T13259 C3INT9 12896796 IC50 > 1000000 nM T13259 C6G5XN 135408704 IC50 > 1000000 nM T13259 D00LMG 5281697 IC50 = 7200000 nM T13259 D03VZF 18169 IC50 = 33100 nM T13259 D07ZBH 97472 IC50 > 1000000 nM T13259 D0L7RB 16036927 IC50 = 350 nM T81900 D05AFR 54682938 IC50 = 100000 nM T81900 D05UBX 42008 IC50 = 7000 nM T81900 D0KL4J 5029 IC50 = 11000 nM T81900 D0B1FE 3194 IC50 = 14 nM T81900 C1FNQ2 53378106 IC50 = 2900 nM T81900 CCKN08 53378322 IC50 > 100000 nM T81900 CGH0S7 54589400 IC50 = 100 nM T81900 C5AG0X 67421743 IC50 > 100000 nM T81900 CV9Q6E 67422054 IC50 = 1400 nM T81900 C0TV7L 67422343 IC50 = 600 nM T81900 CNX47W 67422530 IC50 > 100000 nM T81900 CI9UJ4 71297169 IC50 = 600 nM T81900 C8NUZ1 71601194 Ki > 33000 nM T81900 C1U0FV 71601333 Ki = 25.9 nM T81900 CSN40J 71601334 Ki = 103 nM T81900 CT93WV 71601335 Ki = 1150 nM T81900 C4UK2J 71601336 Ki > 33000 nM T81900 CQC35J 71601478 Ki = 18000 nM T81900 C5FPT7 71601479 Ki = 498 nM T81900 C1YWP7 71601480 Ki = 7750 nM T81900 CW3Y0C 71601481 Ki = 7020 nM T81900 COFN07 71601482 Ki > 33000 nM T81900 C32UCI 71601627 Ki > 33000 nM T81900 CWD10J 71601628 Ki = 87 nM T81900 C4E9HB 71601629 Ki = 5280 nM T81900 C9VDT4 71716848 Ki = 85.1 nM T81900 C5BOQ6 71717486 Ki = 1.4 nM T81900 C6RG8U 71717487 Ki = 73.3 nM T81900 C8BSR4 71718080 Ki = 49.8 nM T81900 C6L3OW 71719891 Ki = 78 nM T81900 CWP5T1 71720518 Ki = 1.7 nM T81900 CMBG30 78318176 IC50 = 56 nM T81900 CO4PK1 91758793 IC50 = 50 nM T81900 C86RXU 155545356 IC50 = 56 nM T81900 D0N9YP 91801116 IC50 = 4 nM T81900 D0T3PW 5281672 IC50 = 100000 nM T15334 D00JQE 11691871 IC50 = 7 nM T15334 D02XXN 49836058 IC50 = 26 nM T15334 D05SSC 6918540 IC50 = 4100 nM T15334 D07HLS 11556427 IC50 = 17.2 nM T15334 D08VBV 57686716 IC50 = 62 nM T15334 D0L0YG 5280335 IC50 = 11500 nM T15334 D05QXT 46880878 IC50 = 24 nM T15334 D03MAD 6918520 IC50 = 73 nM T15334 D07GDN 159325 IC50 = 3 nM T15334 CE18IM 67271 IC50 = 101000 nM T15334 CYI58D 72185 IC50 = 25000 nM T15334 CM14UO 418965 IC50 = 600 nM T15334 CAHN27 465359 IC50 > 500000 nM T15334 C4N0OC 467398 IC50 = 38000 nM T15334 C24AFC 482532 IC50 = 7000 nM T15334 CC9SW1 1304707 IC50 > 30000 nM T15334 C3RL6P 1316302 IC50 = 88 nM T15334 CFW05G 1333727 IC50 = 240 nM T15334 C15YUR 1333885 IC50 = 6810 nM T15334 CL16NM 1361277 IC50 = 280 nM T15334 CH1A7Z 1362920 IC50 > 10000 nM T15334 CZNT56 1363878 IC50 = 4396 nM T15334 CHAC64 1364626 IC50 = 4230 nM T15334 CE97NC 1369980 IC50 = 470 nM T15334 CC4B6G 1370022 IC50 = 13000 nM T15334 C6Q0SB 2236388 IC50 > 10000 nM T15334 CM3GQ8 3346283 IC50 = 13000 nM T15334 C4ON5I 3770260 IC50 > 500000 nM T15334 CCDI37 3938274 IC50 = 4570 nM T15334 C10LPI 4021147 IC50 = 2150 nM T15334 C8YJ9T 4419820 IC50 > 30000 nM T15334 CFP17W 4527804 IC50 > 32000 nM T15334 C2NP4S 5168184 IC50 > 30000 nM T15334 CA73ZW 5283564 IC50 = 65600 nM T15334 CA3MB1 5353801 IC50 = 6300 nM T15334 CFQ3U7 6918766 IC50 = 2000 nM T15334 CZWE38 6918816 IC50 = 3000 nM T15334 C21QRE 7325887 IC50 = 140 nM T15334 CC2UD8 9806610 IC50 = 100 nM T15334 C4ZJ8I 9823684 IC50 = 2000 nM T15334 CV4D8X 9828869 IC50 = 20 nM T15334 CF31MP 9829416 IC50 = 30 nM T15334 C1DMN7 9850223 IC50 > 190000 nM T15334 CYUD89 9863666 IC50 = 1500 nM T15334 CZS3N2 9870704 IC50 = 140 nM T15334 CJ9S4R 9894320 IC50 = 30 nM T15334 CK26LY 9916392 IC50 = 7700 nM T15334 C8YTA7 9935853 IC50 = 20000 nM T15334 CYH50D 9936334 IC50 = 31 nM T15334 C9NMY2 9936855 IC50 = 60.26 nM T15334 CXAH35 9970068 IC50 = 40000 nM T15334 CJ4Z8O 9974016 IC50 = 2000 nM T15334 C56MQN 9977209 IC50 = 4000 nM T15334 CVE0U9 9983064 IC50 = 5000 nM T15334 C3C7AK 9992944 IC50 = 12000 nM T15334 CH4WK3 10002439 IC50 = 13000 nM T15334 C73HEW 10007284 IC50 = 57300 nM T15334 C9YBX6 10031215 IC50 = 195 nM T15334 C7GL0D 10041352 IC50 = 16000 nM T15334 CN05IC 10044138 IC50 = 4000 nM T15334 CT5Q1K 10050438 IC50 = 720 nM T15334 CUDR70 10051680 IC50 = 5000 nM T15334 CIPW54 10053282 IC50 = 86300 nM T15334 CSIK60 10062888 IC50 = 9000 nM T15334 CN5EO3 10073382 IC50 = 1120 nM T15334 CG25TP 10073471 IC50 = 40000 nM T15334 CQVD38 10083422 IC50 = 17000 nM T15334 CKHD08 10088215 IC50 = 72000 nM T15334 CA70OS 10116967 IC50 = 30000 nM T15334 CX2G9R 10119293 IC50 = 70 nM T15334 CAH20E 10120284 IC50 = 90 nM T15334 CA6C3F 10131674 IC50 = 500000 nM T15334 C7GR4H 10142885 IC50 = 200 nM T15334 C48IZL 10144277 IC50 = 100 nM T15334 C9A1JO 10145345 IC50 = 57 nM T15334 CJ2RC0 10162638 IC50 = 23000 nM T15334 C1OT6Q 10164805 IC50 = 90 nM T15334 CBU4V2 10165968 IC50 = 200 nM T15334 CS7A4R 10186806 IC50 = 72000 nM T15334 CLZ58I 10187358 IC50 = 12000 nM T15334 C8E9OA 10188926 IC50 = 60 nM T15334 CMGW21 10208920 IC50 = 49000 nM T15334 CJ7RY9 10216898 IC50 = 3600 nM T15334 CKXT83 10229629 IC50 = 620000 nM T15334 CHFJ90 10229808 IC50 = 30 nM T15334 C92OXJ 10231557 IC50 = 45000 nM T15334 C9G7SR 10232095 IC50 = 29998.53 nM T15334 C8ZOP0 10246927 IC50 = 5000 nM T15334 C02IBR 10281896 IC50 = 190000 nM T15334 CT74EZ 10319013 IC50 = 41000 nM T15334 CMX06G 10319242 IC50 = 60000 nM T15334 C0K5UW 10319633 IC50 = 25000 nM T15334 C9I7WV 10348668 IC50 = 2300 nM T15334 CN69HT 10360154 IC50 = 5000 nM T15334 CRK90Y 10366860 IC50 = 13000 nM T15334 CE4T0K 10430444 IC50 = 61000 nM T15334 CD78MX 10432438 IC50 = 10000 nM T15334 C4B0LM 10434530 IC50 = 4420 nM T15334 CGM64L 10446231 IC50 = 8000 nM T15334 CC5O9G 10498920 IC50 = 15000 nM T15334 CLU9P2 10523012 IC50 = 23000 nM T15334 CV54KL 10549850 IC50 > 500000 nM T15334 CMY14T 10568674 IC50 > 300000 nM T15334 CXLS87 10601339 IC50 = 8000 nM T15334 C2E7GJ 10619814 IC50 > 100000 nM T15334 C7D5LP 10639370 IC50 = 6000 nM T15334 C7L8ST 10648591 IC50 = 5000 nM T15334 C4K0FR 10669141 IC50 = 25000 nM T15334 CB6TX2 10689898 IC50 = 180000 nM T15334 C4CZW1 10691710 IC50 = 41000 nM T15334 C7J5SC 10692165 IC50 = 12000 nM T15334 CFO60Y 10711729 IC50 = 7000 nM T15334 CC3RI0 10721544 IC50 = 4300 nM T15334 C9O7CL 10734409 IC50 = 6000 nM T15334 CC5DT4 10740648 IC50 = 25000 nM T15334 C13AMY 10763332 IC50 = 15000 nM T15334 CKY6R1 10766781 IC50 = 3500 nM T15334 CFR5D4 10769396 IC50 = 3400 nM T15334 CCJI83 10790582 IC50 = 25000 nM T15334 C27AVQ 10804541 IC50 = 7000 nM T15334 C37NMS 10805120 IC50 > 100000 nM T15334 C9QE6O 10806097 IC50 > 100000 nM T15334 CAB70S 10816891 IC50 = 3500 nM T15334 CNXK45 10837030 IC50 > 300000 nM T15334 CJ38PT 10839129 IC50 = 21000 nM T15334 C3RQ2P 10864218 IC50 = 200 nM T15334 C83HBO 10875144 IC50 = 1000 nM T15334 CQ3JH2 10884510 IC50 = 6000 nM T15334 C87TQC 10885641 IC50 > 100000 nM T15334 C8EJM0 10895213 IC50 = 15000 nM T15334 CD6FC9 10895866 IC50 = 1500 nM T15334 CGN27W 10896230 IC50 = 390 nM T15334 CB7KR4 10907408 IC50 = 12000 nM T15334 C96ISB 10918359 IC50 = 3500 nM T15334 CGX3U0 10928074 IC50 = 1000 nM T15334 CBV45K 10940086 IC50 = 1300 nM T15334 CW8J3P 10940406 IC50 = 80 nM T15334 C9LS4Y 10940802 IC50 = 200 nM T15334 C0BEZ2 10948829 IC50 > 100000 nM T15334 CEL51V 10951775 IC50 = 200 nM T15334 C74EUO 10973047 IC50 > 50000 nM T15334 CA9VH0 10973502 IC50 > 50000 nM T15334 C5VUS1 10973830 IC50 = 6900 nM T15334 CKD96A 10984622 IC50 = 100 nM T15334 C3A6BG 10993675 IC50 = 4500 nM T15334 CTL21D 10993963 IC50 = 16000 nM T15334 C1W8SJ 10995194 IC50 = 18000 nM T15334 CHFJ13 11005168 IC50 = 302 nM T15334 CXC8N3 11006225 IC50 = 200 nM T15334 CQ16CK 11006374 IC50 = 2511.89 nM T15334 C2D8UM 11015376 IC50 = 70000 nM T15334 CQHO69 11015903 IC50 = 300 nM T15334 CK2XE1 11017383 IC50 = 400 nM T15334 CP6X9W 11023887 IC50 = 65000 nM T15334 C6LMA8 11038576 IC50 = 1288.25 nM T15334 CFEC07 11039007 IC50 = 400 nM T15334 C1KN4U 11070290 IC50 = 540 nM T15334 COUS34 11071643 IC50 = 80 nM T15334 C8Y7FE 11081883 IC50 = 700 nM T15334 CMR9P6 11082080 IC50 = 300 nM T15334 CG37DS 11091028 IC50 = 15000 nM T15334 CH9Q5M 11091268 IC50 > 50000 nM T15334 C4KY6Q 11092814 IC50 = 400 nM T15334 CINO03 11100897 IC50 > 100000 nM T15334 CKU8Z1 11103994 IC50 = 300 nM T15334 C1U5XG 11113588 IC50 = 50000 nM T15334 CTDJ38 11114287 IC50 = 200 nM T15334 CY9E1T 11124050 IC50 = 2600 nM T15334 C2EAY7 11124385 IC50 = 100 nM T15334 CJO9K2 11124467 IC50 = 500 nM T15334 CEU0V4 11134807 IC50 = 400 nM T15334 CP78AH 11135423 IC50 = 420 nM T15334 C9FBK0 11135705 IC50 = 2400 nM T15334 C9CXI2 11143780 IC50 = 12000 nM T15334 CKH42D 11144753 IC50 = 7800 nM T15334 C63PAC 11145907 IC50 = 80 nM T15334 C2KVA7 11146228 IC50 = 80 nM T15334 CN5FH4 11261706 IC50 = 469 nM T15334 C4TOX2 11498105 IC50 = 14200 nM T15334 C52ROM 11498353 IC50 = 47 nM T15334 CRQE70 11505781 IC50 = 78 nM T15334 C3R5SI 11511556 IC50 = 6000 nM T15334 CYJC54 11513129 IC50 = 20000 nM T15334 C5C3TP 11520198 IC50 = 108 nM T15334 CB25OY 11525926 IC50 = 9000 nM T15334 CJ8A3D 11527073 IC50 = 1430 nM T15334 CC30VP 11527347 IC50 = 13.3 nM T15334 C1UN7A 11527580 IC50 = 365 nM T15334 CVY60T 11527593 IC50 = 66 nM T15334 CK3MV9 11527727 IC50 = 2111 nM T15334 C92TBG 11534811 IC50 = 7815 nM T15334 CT6NC8 11541196 IC50 = 44100 nM T15334 CA9F8M 11541751 IC50 = 753 nM T15334 CBUJ28 11542076 IC50 = 61 nM T15334 CRV0D9 11542316 IC50 = 29 nM T15334 CE13KT 11548962 IC50 = 143 nM T15334 C9LU2N 11554734 IC50 = 23 nM T15334 CD0FW6 11555584 IC50 = 35000 nM T15334 CJNF79 11556473 IC50 = 19.8 nM T15334 CJX85Y 11556603 IC50 = 54 nM T15334 C0PH7J 11561156 IC50 = 11000 nM T15334 CEX1T5 11563293 IC50 = 134 nM T15334 CRMG57 11563741 IC50 = 327 nM T15334 C2CE5Z 11563853 IC50 = 139 nM T15334 CAE9Z2 11570109 IC50 = 46000 nM T15334 CV3UI0 11578015 IC50 = 16.5 nM T15334 C9V6JD 11578460 IC50 = 50000 nM T15334 CJ0I9H 11578475 IC50 = 10100 nM T15334 C5L9TR 11584485 IC50 = 16000 nM T15334 C26VLC 11591906 IC50 = 40000 nM T15334 CK8T1P 11592553 IC50 = 15.2 nM T15334 C1I4AF 11592782 IC50 = 56 nM T15334 C9RKJ6 11592783 IC50 = 40 nM T15334 CGJZ98 11592883 IC50 = 5731 nM T15334 CE31DW 11600044 IC50 = 66 nM T15334 CN8T0G 11600050 IC50 = 15 nM T15334 CQM3A2 11606952 IC50 = 854 nM T15334 CK1YM5 11607128 IC50 = 23 nM T15334 CB4V9F 11607185 IC50 = 151 nM T15334 C7X5LD 11613843 IC50 = 224 nM T15334 C3Y9XP 11614021 IC50 = 296.4 nM T15334 CCAE78 11614176 IC50 = 108 nM T15334 CO1H5D 11614476 IC50 = 36 nM T15334 C3UZL8 11614517 IC50 = 187 nM T15334 CE6HL4 11614539 IC50 = 58 nM T15334 CE7VT2 11621555 IC50 = 1110 nM T15334 CHRL62 11621756 IC50 = 44 nM T15334 C0KSU7 11621765 IC50 = 61 nM T15334 CRUP06 11628674 IC50 = 24.8 nM T15334 C8O6EN 11629007 IC50 = 488 nM T15334 C4CW3K 11629008 IC50 = 72 nM T15334 CUB2F4 11635877 IC50 = 29 nM T15334 CW41RX 11635963 IC50 = 7416 nM T15334 C0U6JA 11648635 IC50 = 45000 nM T15334 CT08IR 11649992 IC50 = 16.7 nM T15334 C5MGK6 11650234 IC50 = 16.2 nM T15334 CZ2E8K 11650398 IC50 = 4555 nM T15334 C6PV8J 11650505 IC50 = 4420 nM T15334 CDB43J 11650506 IC50 = 3790 nM T15334 CH3NG9 11657242 IC50 = 444 nM T15334 CTUG09 11657340 IC50 = 54.1 nM T15334 CL7U8I 11657603 IC50 = 74 nM T15334 CWA43D 11657642 IC50 > 50000 nM T15334 CJC83P 11657764 IC50 = 2915 nM T15334 COYS46 11664298 IC50 = 25 nM T15334 CIN68H 11664694 IC50 = 44 nM T15334 CQ2O4T 11670709 IC50 = 21000 nM T15334 C06KMQ 11671647 IC50 = 133 nM T15334 C06CNB 11671901 IC50 = 5220 nM T15334 C1DMA5 11671961 IC50 = 572 nM T15334 CNDM38 11672080 IC50 = 218 nM T15334 CLM81E 11678430 IC50 = 4664 nM T15334 C29DSU 11686150 IC50 = 16 nM T15334 COTH41 11686285 IC50 = 2350 nM T15334 CLO0D4 11691132 IC50 = 12000 nM T15334 COE2D7 11693067 IC50 = 5700 nM T15334 C4C3FI 11699733 IC50 = 1601 nM T15334 CP1HF6 11699920 IC50 = 210 nM T15334 C0ROE9 11700119 IC50 = 117 nM T15334 C5RK4W 11700350 IC50 = 15 nM T15334 CT0NV7 11706999 IC50 = 23.3 nM T15334 C74CHY 11707240 IC50 = 232 nM T15334 COJ6L9 11707285 IC50 = 3420 nM T15334 CD7Q2B 11714346 IC50 = 23 nM T15334 CY8CK2 11714484 IC50 = 4400 nM T15334 CS9WO8 11714526 IC50 = 49 nM T15334 CS98EU 11714567 IC50 = 37 nM T15334 CMDS05 11721302 IC50 = 4494 nM T15334 CL4T3K 11721460 IC50 = 2590 nM T15334 CJS8M9 11721583 IC50 = 33.5 nM T15334 C53UYZ 11721642 IC50 = 56 nM T15334 C5QL6G 11729174 IC50 = 15000 nM T15334 CY7S2O 11732991 IC50 = 350 nM T15334 C0W3PM 11733217 IC50 = 660 nM T15334 CQ7PZ8 11733434 IC50 > 100000 nM T15334 CR62ZQ 11733526 IC50 = 5200 nM T15334 CI5A0S 11734064 IC50 = 300 nM T15334 C14AFG 11744628 IC50 = 480 nM T15334 CNW0H6 11760922 IC50 = 20000 nM T15334 C5R2AL 11762635 IC50 = 1000 nM T15334 C5PCW0 11782378 IC50 > 100000 nM T15334 CQ9V8A 11792257 IC50 > 300000 nM T15334 C42HOM 11798517 IC50 = 22000 nM T15334 CMS24K 11810932 IC50 = 10000 nM T15334 CT56VR 11813518 IC50 = 300 nM T15334 C64ZUX 11827642 IC50 = 200 nM T15334 CWK20I 11827734 IC50 = 398.11 nM T15334 CRP48D 12086859 IC50 = 55 nM T15334 CK48NC 12086860 IC50 = 70 nM T15334 C7XUZ9 13855380 IC50 = 196000 nM T15334 CZA87M 14331917 IC50 = 46800 nM T15334 CL5JD4 15187131 IC50 > 50000 nM T15334 C8XP4N 15995540 IC50 = 690 nM T15334 CVS58B 16112837 IC50 = 1200 nM T15334 C7CYQ2 16113993 IC50 = 31 nM T15334 C62ASF 16126838 IC50 = 1994 nM T15334 CV03GF 16739908 IC50 = 430 nM T15334 CL5XT8 16739945 IC50 = 90 nM T15334 CBR95H 16739953 IC50 = 6.9 nM T15334 CJ5VL8 16740005 IC50 = 23 nM T15334 CWL04F 16740078 IC50 = 14460 nM T15334 C4VBU0 16743403 IC50 = 2000 nM T15334 C78NVU 16743583 IC50 = 11000 nM T15334 C5NFD2 16743759 IC50 = 200 nM T15334 C19CRM 16743760 IC50 = 12000 nM T15334 C3C7WZ 16743929 IC50 = 4200 nM T15334 C5NU0W 16744101 IC50 = 700 nM T15334 CV7RT1 16744102 IC50 = 400 nM T15334 CWTF57 16744103 IC50 = 7500 nM T15334 C9SN1P 16744104 IC50 = 500 nM T15334 CK28QT 16744269 IC50 = 32000 nM T15334 CG9IY2 16744270 IC50 = 20200 nM T15334 CU3HD2 16744271 IC50 = 12200 nM T15334 CELH12 16744424 IC50 = 1100 nM T15334 C0KX6D 16744425 IC50 = 10800 nM T15334 CRQ72L 16744426 IC50 = 40 nM T15334 CO75DJ 16744595 IC50 = 40 nM T15334 CY1JK2 16744596 IC50 = 100 nM T15334 CLY57P 16744597 IC50 = 20 nM T15334 CA68OS 16744599 IC50 = 14800 nM T15334 CUI0X4 16744748 IC50 = 40 nM T15334 CM3OV0 16745085 IC50 = 90 nM T15334 C94MKR 16745086 IC50 = 50 nM T15334 C5GY6N 16745241 IC50 = 40 nM T15334 C8TKD5 17754437 IC50 = 26 nM T15334 C2XD9E 17754439 IC50 = 39 nM T15334 C59HPD 21157870 IC50 = 22000 nM T15334 CD0P1A 21301191 IC50 = 10000 nM T15334 CO28SL 22956275 IC50 > 300000 nM T15334 CK82HF 22956277 IC50 > 300000 nM T15334 CFPW36 22956278 IC50 = 78000 nM T15334 C1GS0R 22956279 IC50 = 70000 nM T15334 CBP43C 22956282 IC50 > 300000 nM T15334 CWJ5F4 22956283 IC50 > 300000 nM T15334 CKRL72 22956284 IC50 > 300000 nM T15334 C6S8ZY 22956287 IC50 = 40000 nM T15334 C4FGS2 22956371 IC50 = 28000 nM T15334 CXF53Y 23506009 IC50 = 4080 nM T15334 CC03FG 23506029 IC50 = 6720 nM T15334 CC7HD3 23506031 IC50 = 6790 nM T15334 CG49BU 23506040 IC50 = 910 nM T15334 CW7IK8 23506091 IC50 = 45800 nM T15334 CZ09XL 23506103 IC50 = 22900 nM T15334 CNP85A 24738038 IC50 = 91 nM T15334 CT7D9M 24738039 IC50 = 8132 nM T15334 CDI32N 24738196 IC50 = 474 nM T15334 CDN9W7 24738200 IC50 = 254 nM T15334 CL5U2V 24738360 IC50 = 336 nM T15334 CW07RF 24738522 IC50 = 228 nM T15334 CH34GV 24738524 IC50 = 84 nM T15334 C7ZFH2 24738526 IC50 = 1100 nM T15334 CCR35O 24738687 IC50 = 28000 nM T15334 CF8I0D 24739987 IC50 = 1300 nM T15334 CE1H8S 24767813 IC50 = 360 nM T15334 CBYI20 24767814 IC50 = 490 nM T15334 CEC19K 24767818 IC50 = 190 nM T15334 C01SAX 24767824 IC50 = 322 nM T15334 CMVY46 24767828 IC50 = 580 nM T15334 CGF8E2 24767838 IC50 = 45 nM T15334 CZ98XC 24767839 IC50 = 107 nM T15334 C4CJ3D 24767841 IC50 = 271 nM T15334 CV4H3A 24767852 IC50 = 129 nM T15334 C46CKW 24767857 IC50 = 147 nM T15334 CO36XJ 24767858 IC50 = 88 nM T15334 C2KN9O 24767872 IC50 = 560 nM T15334 C6S2VM 24767876 IC50 = 214 nM T15334 CJ86YX 24767890 IC50 = 133 nM T15334 C8F0IY 24767892 IC50 = 50 nM T15334 C9B2NX 24767901 IC50 = 14 nM T15334 C4J9RW 24767903 IC50 = 94 nM T15334 CY3W2H 24767905 IC50 = 41 nM T15334 C7SLF3 24774836 IC50 = 33 nM T15334 CVPW54 24774923 IC50 = 500 nM T15334 CAZK91 24774924 IC50 = 235 nM T15334 CLZM20 24774925 IC50 = 117 nM T15334 C9UN5H 24774926 IC50 = 64 nM T15334 CW4Y0D 24774927 IC50 = 143 nM T15334 CJ6U8D 24775099 IC50 = 125 nM T15334 C5B9EO 24775283 IC50 = 326 nM T15334 CQ57RB 24775284 IC50 = 744 nM T15334 CLUX04 24775285 IC50 = 331 nM T15334 CKI5W8 24775382 IC50 = 125 nM T15334 CUZQ92 24775565 IC50 = 277000 nM T15334 CY3X0K 24775566 IC50 = 345000 nM T15334 CV9FA1 24775568 IC50 = 126 nM T15334 C1LIO0 24775653 IC50 = 317000 nM T15334 C4WC8O 24775654 IC50 > 3000 nM T15334 CU3RE2 24775745 IC50 = 600 nM T15334 C5CHT0 24775748 IC50 = 96 nM T15334 CISJ85 25010200 IC50 = 10 nM T15334 CRI29V 25108841 IC50 = 22 nM T15334 C5Q6GA 25108843 IC50 = 67 nM T15334 CYOV03 25150901 IC50 = 154 nM T15334 CMS9R3 25151607 IC50 = 40 nM T15334 C0XBY4 25151662 IC50 = 19160 nM T15334 CD70KZ 25151793 IC50 = 78 nM T15334 CHU1R7 25151849 IC50 = 46 nM T15334 C7XDZ8 25151850 IC50 = 140 nM T15334 CC1T8M 25151988 IC50 = 133 nM T15334 CH9NA3 25151989 IC50 = 84 nM T15334 C5AY6K 25151990 IC50 = 37 nM T15334 C05HFO 25152653 IC50 = 171 nM T15334 C8HXD1 25152860 IC50 = 124 nM T15334 C7N4FW 25152862 IC50 = 2342 nM T15334 CXC85P 25153077 IC50 = 829 nM T15334 CZI56N 25153212 IC50 = 77 nM T15334 CJW29T 25153282 IC50 = 955 nM T15334 CR0EH4 25153700 IC50 = 66 nM T15334 C69DRY 25169787 IC50 = 40 nM T15334 CEY30L 25170006 IC50 = 306 nM T15334 C40YPZ 25170007 IC50 = 114 nM T15334 CC03WI 25170008 IC50 = 61 nM T15334 CLO9E2 25170009 IC50 = 37 nM T15334 CC4K8E 25170211 IC50 = 223 nM T15334 CXG80Q 25170213 IC50 = 114 nM T15334 C15NAH 25170415 IC50 = 43 nM T15334 CYQ2X5 25170416 IC50 = 13 nM T15334 C0XM1F 25170417 IC50 = 31 nM T15334 C8JZF0 25170418 IC50 = 19 nM T15334 CKTF27 25172077 IC50 = 300 nM T15334 CIM85L 25172282 IC50 = 131 nM T15334 C5Q8YH 25172671 IC50 = 243 nM T15334 CJ40GB 44288699 IC50 = 3960 nM T15334 CH9N3V 44288890 IC50 = 15000 nM T15334 C5N2YC 44289347 IC50 = 6240 nM T15334 CRM9X0 44289349 IC50 = 14300 nM T15334 C96NUW 44301393 IC50 = 6000 nM T15334 C5WF1Y 44301411 IC50 = 15000 nM T15334 CE58LZ 44301412 IC50 = 24000 nM T15334 CRN6S9 44301418 IC50 = 5000 nM T15334 CFR6C8 44301622 IC50 = 14000 nM T15334 CTWY93 44303460 IC50 = 4300 nM T15334 CHW7I2 44303461 IC50 = 6900 nM T15334 CH65FG 44303582 IC50 = 5200 nM T15334 C9WQ1U 44303597 IC50 > 50000 nM T15334 C32HSP 44303605 IC50 > 50000 nM T15334 C7FLW5 44303606 IC50 = 46000 nM T15334 CY1SA0 44303666 IC50 = 34000 nM T15334 CT2H0B 44303817 IC50 = 25000 nM T15334 CZH2I1 44303838 IC50 = 18000 nM T15334 CZX56S 44303890 IC50 = 47000 nM T15334 C3CZQ6 44321273 IC50 = 102000 nM T15334 C4I1BJ 44370883 IC50 = 46000 nM T15334 C73UKI 44371111 IC50 = 23000 nM T15334 CVX3H5 44382873 IC50 = 11000 nM T15334 C07IUS 44383661 IC50 = 9000 nM T15334 CA0V7G 44397737 IC50 = 1500 nM T15334 C0KFR3 44397738 IC50 = 200 nM T15334 CKW30I 44397750 IC50 = 4000 nM T15334 C9QYH4 44397766 IC50 = 30 nM T15334 C3C4UL 44397769 IC50 = 15 nM T15334 CP28HX 44397791 IC50 = 200 nM T15334 C9YC8P 44397795 IC50 = 13000 nM T15334 CG8VK0 44397796 IC50 = 200 nM T15334 CHUW43 44397824 IC50 = 10000 nM T15334 C6TD7Q 44397825 IC50 = 800 nM T15334 CZ60RG 44397833 IC50 = 10000 nM T15334 C6TD7H 44397850 IC50 = 2000 nM T15334 CA79UJ 44397851 IC50 = 600 nM T15334 CZB5S8 44397854 IC50 = 60 nM T15334 C47ICW 44397864 IC50 = 700 nM T15334 CSI8B7 44397881 IC50 = 30 nM T15334 CZC39D 44397886 IC50 > 20000 nM T15334 CXME59 44397896 IC50 = 400 nM T15334 CAJO76 44397899 IC50 > 20000 nM T15334 C5LN6Y 44397900 IC50 = 200 nM T15334 C0SM7L 44397930 IC50 = 3000 nM T15334 CKJ82B 44397950 IC50 = 4000 nM T15334 CBO3R0 44397953 IC50 = 1500 nM T15334 C0UWO6 44397967 IC50 = 6000 nM T15334 CA61BG 44397970 IC50 = 800 nM T15334 C6JQC9 44397983 IC50 = 32 nM T15334 C92JAS 44397985 IC50 > 20000 nM T15334 C5P7AN 44397994 IC50 = 700 nM T15334 CF3D4Y 44435686 IC50 = 30 nM T15334 C6XDL8 44435688 IC50 = 200 nM T15334 C2SY6B 44435692 IC50 = 60 nM T15334 CU6G8V 44435705 IC50 = 4080 nM T15334 C57AGV 44435706 IC50 = 6720 nM T15334 C2YQG0 44435707 IC50 = 15000 nM T15334 C9ACQ0 44435709 IC50 = 12000 nM T15334 CQ7W2S 44435710 IC50 = 45800 nM T15334 CT20YG 44435711 IC50 = 89.13 nM T15334 CYHS63 44435713 IC50 = 79.43 nM T15334 CKH8E6 44435714 IC50 = 7762.47 nM T15334 C0TE4B 44435715 IC50 = 6240 nM T15334 C9OB0T 44435717 IC50 = 70 nM T15334 C89SOM 44435725 IC50 = 3630.78 nM T15334 CGZQ74 44439033 IC50 > 100000 nM T15334 C0FYD3 44439035 IC50 > 100000 nM T15334 CNY6I7 44439039 IC50 = 5000 nM T15334 CO3NC5 44439044 IC50 = 1900 nM T15334 C2S0ZW 44439052 IC50 = 93400 nM T15334 C5WBT7 44439054 IC50 = 500 nM T15334 CWPS81 44439081 IC50 = 230 nM T15334 CHL5T4 44439096 IC50 = 62590 nM T15334 CZ7B1S 44439097 IC50 = 100000 nM T15334 CFM9B6 44439100 IC50 = 46380 nM T15334 CE3QV6 44439104 IC50 = 100000 nM T15334 CD1TO8 44439107 IC50 = 100000 nM T15334 CYZL56 44439110 IC50 = 36900 nM T15334 CP27VK 44439115 IC50 = 32500 nM T15334 C7P2LO 44439137 IC50 = 14580 nM T15334 C9J1NB 44439138 IC50 = 2225 nM T15334 CTIR63 44439181 IC50 = 54570 nM T15334 CNY46R 44439184 IC50 = 1500 nM T15334 C2JT6Q 44449749 IC50 = 18000 nM T15334 C39OJY 44449751 IC50 = 56 nM T15334 C8IW5S 44449754 IC50 = 92 nM T15334 CGF31D 44449755 IC50 = 52 nM T15334 CQN3G9 44449772 IC50 = 97 nM T15334 C61HWM 44449774 IC50 = 3500 nM T15334 C9DPZ2 44449779 IC50 = 27000 nM T15334 CE78UH 44449802 IC50 > 32000 nM T15334 CMYC41 44449804 IC50 = 1700 nM T15334 CA13VW 44449805 IC50 = 3500 nM T15334 CW71NA 44449806 IC50 > 32000 nM T15334 C3Q5SY 44449834 IC50 > 32000 nM T15334 CW4R8U 44449835 IC50 > 32000 nM T15334 C2DNU6 44449858 IC50 > 10000 nM T15334 CE8M4K 44449860 IC50 > 32000 nM T15334 CI1N9V 44449861 IC50 > 10000 nM T15334 CFOU56 44449862 IC50 > 32000 nM T15334 CR13XQ 44449863 IC50 > 32000 nM T15334 CCNI21 44449885 IC50 > 10000 nM T15334 CD5V9C 44449889 IC50 > 10000 nM T15334 CIG68Y 44449892 IC50 = 130 nM T15334 CA2DU8 44449916 IC50 > 10000 nM T15334 C4US5J 44449918 IC50 = 31 nM T15334 CJR51B 44449919 IC50 = 23 nM T15334 CW1JR7 44449920 IC50 = 120 nM T15334 CYE72G 44449921 IC50 = 96 nM T15334 CSLO76 44449950 IC50 = 120 nM T15334 CV6IZ5 44449951 IC50 = 590 nM T15334 CEX21A 44449952 IC50 = 200 nM T15334 C2TQ6O 44449953 IC50 = 1200 nM T15334 CN6IW3 44449954 IC50 > 32000 nM T15334 CP7HO6 44449983 IC50 > 10000 nM T15334 CYQ8U9 44449984 IC50 = 3600 nM T15334 CFI16W 44449985 IC50 = 1900 nM T15334 CC24XT 44449986 IC50 = 200 nM T15334 CDBQ78 44450010 IC50 = 2300 nM T15334 C2JW6S 44450011 IC50 > 10000 nM T15334 C5KP6U 44450012 IC50 = 9300 nM T15334 CD4H1P 44450013 IC50 = 3300 nM T15334 C06KTQ 44450014 IC50 = 11000 nM T15334 CJD04O 44450037 IC50 = 32000 nM T15334 CIT90V 44450038 IC50 > 10000 nM T15334 C12UVS 44450039 IC50 = 900 nM T15334 C1E2GN 44450040 IC50 = 1900 nM T15334 CX9Z5N 44450041 IC50 > 32000 nM T15334 CW5XF1 44450042 IC50 > 32000 nM T15334 C1RY3G 44450043 IC50 > 32000 nM T15334 CE2S4J 44450062 IC50 > 10000 nM T15334 C0L1ED 44450066 IC50 = 220 nM T15334 C23ILE 44450067 IC50 > 10000 nM T15334 CXQL65 44450068 IC50 > 32000 nM T15334 CG1O9U 44450069 IC50 > 32000 nM T15334 CY0O1J 44450098 IC50 = 380 nM T15334 CR4NW2 44450099 IC50 = 1300 nM T15334 C3EQ7J 44450126 IC50 = 11 nM T15334 CUW83L 44450127 IC50 = 18 nM T15334 C7B0XR 44450128 IC50 > 10000 nM T15334 C81SNP 44450129 IC50 = 15 nM T15334 CX14MA 44450130 IC50 > 10000 nM T15334 C9NRC7 44450131 IC50 = 8300 nM T15334 CV37RN 44450162 IC50 = 85 nM T15334 C4LT7A 44450164 IC50 = 18 nM T15334 CZN93T 44450165 IC50 > 10000 nM T15334 CXIR61 44450166 IC50 > 10000 nM T15334 CF50SL 44450167 IC50 = 1100 nM T15334 CR1G2A 44450168 IC50 = 7300 nM T15334 CGB1X9 44450191 IC50 = 40 nM T15334 CA1M7Y 44450192 IC50 = 42 nM T15334 CMD45W 44450194 IC50 > 10000 nM T15334 CS8JQ4 44593732 IC50 = 400 nM T15334 CAR13E 46216790 IC50 = 151 nM T15334 CK6CU5 46226907 IC50 = 28 nM T15334 C6Y2RS 46230594 IC50 > 30000 nM T15334 C9XEW2 46230595 IC50 = 1774 nM T15334 CRN4X0 46230596 IC50 = 2206 nM T15334 C2YA5I 46230624 IC50 = 6537 nM T15334 C6N0OC 46230625 IC50 = 18080 nM T15334 CLK28T 46230626 IC50 > 30000 nM T15334 CTY65E 46230627 IC50 > 30000 nM T15334 CMC79V 46230675 IC50 > 30000 nM T15334 C34KBX 46230676 IC50 > 30000 nM T15334 C58QAY 46230677 IC50 > 30000 nM T15334 CA8TN4 46230678 IC50 > 30000 nM T15334 C8P1LF 46230725 IC50 = 1182 nM T15334 CQBT61 46230726 IC50 = 505 nM T15334 CVQ6Z5 46230727 IC50 = 1375 nM T15334 COM79U 46230728 IC50 = 613 nM T15334 CP5X0W 46230787 IC50 = 132 nM T15334 C7P6NW 46230788 IC50 = 94 nM T15334 C80NSW 46230789 IC50 = 51 nM T15334 C46ABD 46230790 IC50 = 151 nM T15334 C4I2HK 46230791 IC50 = 75900 nM T15334 C60AQU 46230837 IC50 = 890 nM T15334 C1G3JS 46231048 IC50 = 44 nM T15334 C7OS5C 46231106 IC50 = 2587 nM T15334 C8QB6L 46231107 IC50 = 2700 nM T15334 C6FGS1 46231108 IC50 = 6390 nM T15334 C80KQM 46231179 IC50 > 30000 nM T15334 CN38YR 46231180 IC50 > 30000 nM T15334 CVZ8G7 46231181 IC50 > 30000 nM T15334 C54AIN 46231182 IC50 = 19310 nM T15334 CWK83Y 46231238 IC50 = 1773 nM T15334 CHM6S2 46231239 IC50 = 1248 nM T15334 CU45IW 46231280 IC50 > 30000 nM T15334 C9KH1N 46231281 IC50 = 12880 nM T15334 C0H1TD 46231282 IC50 = 26490 nM T15334 CHR6Q1 46231326 IC50 = 810 nM T15334 CUB6G2 46232843 IC50 = 193 nM T15334 CY97JH 46865658 IC50 = 17 nM T15334 CT7IH6 46880281 IC50 = 60 nM T15334 C1EZ0I 46880282 IC50 = 2000 nM T15334 CI69ZS 46880283 IC50 = 3000 nM T15334 CX6J8D 46880319 IC50 = 15000 nM T15334 CS4VX6 46880320 IC50 > 20000 nM T15334 C29HUP 46880321 IC50 = 500 nM T15334 C0HC3V 46880322 IC50 > 20000 nM T15334 CJ0K6M 46880323 IC50 = 15000 nM T15334 CD3JL1 46880360 IC50 = 4000 nM T15334 C7WZE9 46880361 IC50 = 80 nM T15334 CUI35G 46880362 IC50 = 100 nM T15334 CM2Y4O 46880363 IC50 = 70 nM T15334 CZ65HQ 46880406 IC50 = 100 nM T15334 C94SNM 46880459 IC50 = 22 nM T15334 CQ79ZH 46880460 IC50 = 39 nM T15334 C27KLC 46880879 IC50 = 4500 nM T15334 CAF18V 46880880 IC50 = 600 nM T15334 C9FK5G 46880926 IC50 = 2000 nM T15334 C2DIV5 46880927 IC50 = 600 nM T15334 C7B8OE 46880928 IC50 = 300 nM T15334 CYUC84 46880929 IC50 = 3000 nM T15334 CB49OT 46880965 IC50 = 90 nM T15334 CUE79T 46880966 IC50 = 70 nM T15334 CI81ZS 46880967 IC50 = 33 nM T15334 C83MVG 46905196 IC50 = 19700 nM T15334 CDK39J 49864871 IC50 = 30000 nM T15334 CUMW31 49864908 IC50 = 25000 nM T15334 CPI7U5 49864910 IC50 = 25000 nM T15334 CTIM49 50925393 IC50 = 1725 nM T15334 CQE3M0 50941639 IC50 = 13 nM T15334 CCXI27 50941728 IC50 = 16 nM T15334 CJH80D 51346897 IC50 = 22 nM T15334 C2LMK0 52941282 IC50 = 3832 nM T15334 CJBP56 52941413 IC50 = 9514 nM T15334 C70BVA 52945032 IC50 = 694 nM T15334 CJP20Y 53248833 IC50 = 93 nM T15334 CZT58S 53316779 IC50 = 40 nM T15334 CEX5P9 53316824 IC50 > 30000 nM T15334 CW04QB 53316825 IC50 = 382 nM T15334 C5WC8B 53316826 IC50 = 625 nM T15334 CAN10H 53316827 IC50 = 207 nM T15334 CA4L2W 53316828 IC50 = 64 nM T15334 C4KQ0N 53317008 IC50 = 3186 nM T15334 CS0J5M 53317084 IC50 > 10000 nM T15334 CE2B0I 53317085 IC50 > 10000 nM T15334 CM4KP9 53317086 IC50 = 229 nM T15334 CGM53I 53317107 IC50 = 2172 nM T15334 CP4QL9 53317108 IC50 = 5741 nM T15334 C2S3IU 53318321 IC50 = 2742 nM T15334 CT61CB 53318372 IC50 = 47 nM T15334 C5NJG0 53318373 IC50 = 28 nM T15334 CUP5Q2 53318374 IC50 = 29 nM T15334 CW5K7D 53319022 IC50 = 287 nM T15334 C6LWJ4 53319231 IC50 = 58 nM T15334 CD4Q0L 53319415 IC50 = 53 nM T15334 CSB91R 53319484 IC50 = 115 nM T15334 CHB62C 53319709 IC50 = 39 nM T15334 CP2NX9 53320329 IC50 = 221 nM T15334 CV72DL 53320717 IC50 = 111 nM T15334 C6KA8T 53320718 IC50 = 9164 nM T15334 C4VC2Y 53320782 IC50 = 92 nM T15334 CI6BC7 53320783 IC50 = 72 nM T15334 C36JGT 53320784 IC50 = 83 nM T15334 C83XBM 53320945 IC50 = 2612 nM T15334 CXBS43 53321463 IC50 = 4554 nM T15334 CM2E9L 53321660 IC50 = 8940 nM T15334 C15QYV 53322008 IC50 = 19 nM T15334 C7EOI3 53322009 IC50 = 65 nM T15334 C5ZI6B 53322089 IC50 = 130 nM T15334 CRQ17W 53322090 IC50 = 951 nM T15334 C3AML5 53322091 IC50 = 356 nM T15334 CSR03V 53322362 IC50 = 975 nM T15334 CVX56R 53322363 IC50 = 2053 nM T15334 CB9PO0 53322364 IC50 = 4029 nM T15334 CVU37M 53322970 IC50 = 31 nM T15334 CRZH65 53322977 IC50 = 146 nM T15334 C1FV9P 53322981 IC50 = 99 nM T15334 CPMB72 53323366 IC50 > 30000 nM T15334 CTCN81 53323367 IC50 = 49 nM T15334 CNR7J6 53323368 IC50 = 99 nM T15334 C4KV3M 53323369 IC50 > 30000 nM T15334 CFS3L9 53323443 IC50 = 111 nM T15334 CB3G9A 53323689 IC50 = 110 nM T15334 CH37UZ 53323704 IC50 = 48 nM T15334 CG16WS 53323705 IC50 = 24 nM T15334 CJL9M0 53323706 IC50 = 413 nM T15334 CX5E9M 53324688 IC50 = 69 nM T15334 CJ7N5D 53324948 IC50 = 18760 nM T15334 CX3JI0 53325001 IC50 = 15 nM T15334 CRT7Z9 53325002 IC50 = 2249 nM T15334 CYB47G 53325995 IC50 = 64 nM T15334 CS61DY 53326049 IC50 = 280 nM T15334 CJM7V0 53326050 IC50 = 256 nM T15334 CP9BE1 53326205 IC50 = 198 nM T15334 CJA7H9 53326237 IC50 = 11600 nM T15334 C08UNO 53326803 IC50 = 1253 nM T15334 CO92DK 53326840 IC50 = 874 nM T15334 CQ7LB1 53327841 IC50 = 22 nM T15334 CC6ME0 53327888 IC50 = 18 nM T15334 CDA2S6 53363909 IC50 = 25.6 nM T15334 C2D5CN 53363910 IC50 = 39.3 nM T15334 CF3ER8 53363911 IC50 = 5670 nM T15334 CY51UW 53363996 IC50 = 266 nM T15334 CFC07T 53363998 IC50 = 268 nM T15334 C3D4XR 53364079 IC50 = 17.8 nM T15334 CL8U1F 53467539 IC50 = 51 nM T15334 CKA5R3 53467746 IC50 = 1433 nM T15334 C04YEO 53467748 IC50 = 548 nM T15334 C3CT2Q 53467749 IC50 = 45 nM T15334 CR2ON7 53467960 IC50 = 37 nM T15334 C78QOS 53467962 IC50 = 796 nM T15334 CQ6K5V 53467965 IC50 = 29 nM T15334 CBV76D 53468189 IC50 = 42 nM T15334 CR50JO 53468402 IC50 = 1077 nM T15334 CLI3M4 53468403 IC50 = 96 nM T15334 C4BL3X 53468405 IC50 = 47 nM T15334 CF29ME 53468599 IC50 = 131 nM T15334 CP5O7F 53468799 IC50 = 18 nM T15334 C3NC0Q 53469197 IC50 = 418 nM T15334 CA6V9P 53469394 IC50 = 524 nM T15334 C65HGY 57390584 IC50 = 27.1 nM T15334 CEU47T 57390685 IC50 = 18 nM T15334 C5EMC8 57390686 IC50 = 6935 nM T15334 CEY18F 57391801 IC50 = 37200 nM T15334 CLWZ01 57392491 IC50 = 19.6 nM T15334 CNT2W7 57394193 IC50 = 24.9 nM T15334 C6IG9Z 57394194 IC50 = 254.2 nM T15334 C14ONF 57395247 IC50 = 27300 nM T15334 C08RLC 57395961 IC50 = 23.5 nM T15334 CWM92X 57397757 IC50 = 1229 nM T15334 CKOX28 57397758 IC50 = 689.1 nM T15334 CK5V7G 57397759 IC50 = 2599 nM T15334 CE1IF6 57402259 IC50 = 293 nM T15334 CBH7K5 57402946 IC50 = 31.21 nM T15334 C0GY1C 57402947 IC50 = 71.8 nM T15334 CJUA84 57686685 IC50 = 60 nM T15334 C0LY5O 57686707 IC50 = 150 nM T15334 CY0XJ7 57686750 IC50 = 160 nM T15334 C6YUW2 57963381 IC50 = 60 nM T15334 CLC8V7 57963497 IC50 = 71 nM T15334 CF3LU0 57963505 IC50 = 771 nM T15334 CTE3S5 57963518 IC50 = 240 nM T15334 C75BPF 58615273 IC50 = 13 nM T15334 CM5H0D 58897193 IC50 > 32000 nM T15334 CEX25L 58898116 IC50 = 5 nM T15334 CDF36I 58919900 IC50 = 7100 nM T15334 C38TSW 58920059 IC50 = 16 nM T15334 CR7EM4 58920071 IC50 = 85 nM T15334 C87BWE 58920089 IC50 = 50 nM T15334 CGC9W6 58920153 IC50 = 310 nM T15334 C0FY6C 58920163 IC50 = 1 nM T15334 CZ0QU8 58920185 IC50 = 3800 nM T15334 CL1DG9 58920226 IC50 = 130 nM T15334 CMB3Y8 58920230 IC50 = 130 nM T15334 C6UNB5 58920231 IC50 = 1.5 nM T15334 CUG0X4 58920248 IC50 = 5500 nM T15334 CE8LT7 58920275 IC50 = 700 nM T15334 CXF4W9 58920284 IC50 = 35 nM T15334 CC34QG 58920291 IC50 = 9 nM T15334 CCNI49 58920310 IC50 = 120 nM T15334 C2TQ5Y 58920313 IC50 = 26 nM T15334 C01CHS 58920320 IC50 = 620 nM T15334 C5SLZ8 58920342 IC50 = 1100 nM T15334 C4OEH8 58920354 IC50 = 20000 nM T15334 CN57AI 58920359 IC50 = 22 nM T15334 CJ14ZD 58920474 IC50 = 34000 nM T15334 CXGW57 58920485 IC50 = 5900 nM T15334 C7XO4Q 58920527 IC50 = 970 nM T15334 C9CG0T 58920654 IC50 > 96000 nM T15334 C8IN2X 58920676 IC50 = 10000 nM T15334 C84WIB 58920695 IC50 = 6 nM T15334 CPN61O 58920709 IC50 = 6 nM T15334 C0C1SF 58920716 IC50 = 50 nM T15334 CONZ75 58920736 IC50 = 641 nM T15334 CF0AM7 58920741 IC50 = 7 nM T15334 C18XAF 58920742 IC50 = 27000 nM T15334 C56YJS 58920756 IC50 = 27000 nM T15334 CD19AE 58920757 IC50 = 7 nM T15334 CK6F4V 58920821 IC50 = 25 nM T15334 CBH6N7 58920845 IC50 = 52 nM T15334 CKSH46 58920856 IC50 = 24040 nM T15334 CO8N2R 58920867 IC50 = 240 nM T15334 CVY0Q2 58920980 IC50 > 96000 nM T15334 CWR0X1 58921056 IC50 = 170 nM T15334 C21IEH 58921084 IC50 = 2900 nM T15334 CTS7K3 58921113 IC50 = 4230 nM T15334 C1PD2T 58921128 IC50 = 32750 nM T15334 CUE6Z5 58921163 IC50 = 19140 nM T15334 C2PIO0 58921211 IC50 = 36 nM T15334 C94QOD 58921229 IC50 = 520 nM T15334 C40JTS 58921261 IC50 = 20 nM T15334 C1E0SA 58921334 IC50 = 2400 nM T15334 CZU10Y 58921504 IC50 = 31 nM T15334 C58TRS 58921572 IC50 = 3097 nM T15334 CB3NZ6 58921591 IC50 = 33330 nM T15334 CMW7K2 58921607 IC50 = 3300 nM T15334 C51KNJ 58921618 IC50 = 10 nM T15334 C8KV0G 58921650 IC50 = 12000 nM T15334 CZ8J9R 58921651 IC50 = 140 nM T15334 CNM0P2 58921656 IC50 = 8532 nM T15334 CY8MT0 58921738 IC50 = 9 nM T15334 CSOL31 59458454 IC50 = 62 nM T15334 C0L2FW 59458459 IC50 = 3 nM T15334 C83DOJ 59458460 IC50 = 1 nM T15334 C0ZLU4 59458594 IC50 = 2.5 nM T15334 CZ0Q7W 59458647 IC50 = 11 nM T15334 CV41DL 59458714 IC50 = 26 nM T15334 C6K0MO 59458732 IC50 = 1.8 nM T15334 CFP75N 59458738 IC50 = 3300 nM T15334 CT8Z7J 59458907 IC50 = 6 nM T15334 CJ5I3Q 59459021 IC50 = 1.3 nM T15334 C9XI4D 59459390 IC50 = 230 nM T15334 CTH04J 59459492 IC50 = 2.9 nM T15334 C2SNL8 59541239 IC50 = 5 nM T15334 CI8WC3 60148979 IC50 = 14 nM T15334 C7BJ6P 60170170 IC50 = 6700 nM T15334 CK9UF1 60170171 IC50 = 44000 nM T15334 CST03D 60170256 IC50 = 1300 nM T15334 CS3MN8 60170257 IC50 = 1100 nM T15334 CXRF65 60170258 IC50 = 8900 nM T15334 C2B8RC 60170439 IC50 = 36 nM T15334 CNQ9R4 60170524 IC50 = 15 nM T15334 C12IMJ 66762745 IC50 = 135 nM T15334 CT9W7Q 70681157 IC50 > 50000 nM T15334 C32GOA 70681182 IC50 = 591 nM T15334 CN3F1X 70681183 IC50 = 471 nM T15334 CZ96AD 70681685 IC50 = 24 nM T15334 CT1NA4 70681686 IC50 = 48 nM T15334 C83JZM 70683266 IC50 = 1050 nM T15334 CN4JK5 70683267 IC50 > 5000 nM T15334 CK4F9R 70683268 IC50 > 50000 nM T15334 CR4MO6 70683269 IC50 = 142 nM T15334 CUK8Y1 70683273 IC50 = 12 nM T15334 CQ2V1F 70683274 IC50 = 21 nM T15334 C25WJR 70683275 IC50 = 24 nM T15334 CY8A9F 70683276 IC50 = 197 nM T15334 C91RUY 70685367 IC50 = 1297 nM T15334 C40JXB 70685382 IC50 = 25000 nM T15334 CTA0U4 70687507 IC50 = 98 nM T15334 CVK18D 70687515 IC50 = 38.4 nM T15334 C3KI5U 70687516 IC50 = 114 nM T15334 C0KF9W 70687517 IC50 = 193 nM T15334 C2KV3X 70689560 IC50 = 396 nM T15334 CR1SO4 70689561 IC50 = 980 nM T15334 C2J7UR 70689562 IC50 = 74 nM T15334 C46DUR 70689563 IC50 = 47 nM T15334 C91NZC 70689577 IC50 > 50000 nM T15334 C9LT1D 70689578 IC50 = 825 nM T15334 COE6V9 70689911 IC50 = 162 nM T15334 CX70ZK 70690095 IC50 = 47 nM T15334 CQ2WS7 70691703 IC50 = 30 nM T15334 CXY0C2 70691704 IC50 = 55 nM T15334 CB3NQ6 70691705 IC50 = 205 nM T15334 CXQ61L 70692254 IC50 = 2310 nM T15334 CRJ1C7 70692255 IC50 = 42 nM T15334 CQM53F 70693768 IC50 = 948 nM T15334 CKB26E 70693769 IC50 = 203 nM T15334 CKXQ64 70693770 IC50 = 154 nM T15334 CH7WD2 70693771 IC50 = 134 nM T15334 C45OFZ 70693772 IC50 = 31 nM T15334 CMK9A0 70693784 IC50 = 20 nM T15334 CKU30X 70694323 IC50 = 26 nM T15334 CO32ZA 70694324 IC50 = 55 nM T15334 CTQW74 70695882 IC50 = 487 nM T15334 C8O0PW 70695883 IC50 = 980 nM T15334 CGL2Z1 70695893 IC50 = 106 nM T15334 C5E6CR 70695894 IC50 = 24 nM T15334 CR14VD 70695895 IC50 = 207 nM T15334 CDQ24L 71451229 IC50 = 27 nM T15334 CMC4R0 71453045 IC50 = 1740 nM T15334 CXL81R 71453441 IC50 = 6900 nM T15334 CMY06A 71454788 IC50 = 91820 nM T15334 CCH1G9 71456563 IC50 = 44590 nM T15334 C7YV5S 71460260 IC50 = 1270 nM T15334 CUQ36S 71460261 IC50 = 2 nM T15334 C31GKZ 71532592 IC50 = 20 nM T15334 COA7X9 71532660 IC50 = 11 nM T15334 C7H3VA 71580010 IC50 = 23100 nM T15334 CG5BJ2 71580539 IC50 = 68500 nM T15334 C34MKE 73350199 IC50 = 300 nM T15334 C24ZFJ 76310713 IC50 = 40 nM T15334 C6FO9E 87152177 IC50 = 140 nM T15334 CPNF83 91669216 IC50 = 94 nM T15334 C1S4DM 118007876 IC50 = 8958 nM T15334 C5RV9Y 118007916 IC50 = 937 nM T15334 CDSY89 118007954 IC50 = 1218 nM T15334 CO52AP 118007960 IC50 = 917 nM T15334 C1LH3U 118007971 IC50 = 308 nM T15334 CPLC19 118007995 IC50 = 1375 nM T15334 C62JTW 118014018 IC50 = 1996 nM T15334 CG9IW3 118014038 IC50 = 101 nM T15334 CS84UA 118014260 IC50 = 763 nM T15334 CZWA98 118014261 IC50 = 232 nM T15334 C8PF2J 118014262 IC50 = 9683 nM T15334 C1RGI5 118014264 IC50 = 222 nM T15334 C6BZA5 118014266 IC50 = 69 nM T15334 C07TMF 118014267 IC50 = 491 nM T15334 CK27HE 118014275 IC50 = 3374 nM T15334 C1IET2 118014279 IC50 = 2602 nM T15334 C9LIA2 118014302 IC50 = 746 nM T15334 C28TXI 118723757 IC50 = 4052 nM T15334 C3GKX9 118724180 IC50 = 576 nM T15334 C4OMY5 124603198 IC50 = 60 nM T15334 C53NIT 126695273 IC50 = 150 nM T15334 CG7VZ9 126695276 IC50 = 690 nM T15334 C41XMR 126695292 IC50 = 5200 nM T15334 CNY7R5 126695294 IC50 = 14200 nM T15334 CVH7F6 126695297 IC50 = 29600 nM T15334 CW5AY3 126695302 IC50 = 2000 nM T15334 CZV5B7 126695321 IC50 > 50000 nM T15334 C4SFW1 127026267 IC50 = 2900 nM T15334 CVH0O9 127026270 IC50 = 6700 nM T15334 CYQ14J 127026271 IC50 = 240 nM T15334 CJ8RO1 127026560 IC50 = 5400 nM T15334 C9MNK5 127026561 IC50 = 9500 nM T15334 C3O5VW 127026562 IC50 = 3500 nM T15334 C02MKP 127026564 IC50 = 18200 nM T15334 CLVY21 127026565 IC50 = 2800 nM T15334 CZO0C4 127026566 IC50 = 9100 nM T15334 CZQ5Y7 127026567 IC50 = 16700 nM T15334 CVL03N 127026568 IC50 = 2700 nM T15334 CA1Q8P 127026569 IC50 = 1300 nM T15334 CX4OG7 127026570 IC50 = 3400 nM T15334 C6QTC1 127026571 IC50 = 2300 nM T15334 CH62UP 127026572 IC50 > 50000 nM T15334 CA4I5M 127032509 IC50 = 37800 nM T15334 CG1QE5 127032510 IC50 = 11300 nM T15334 CCA08Y 127032511 IC50 = 19500 nM T15334 CE8A0X 127033402 IC50 = 11800 nM T15334 CNM2H5 127033403 IC50 > 50000 nM T15334 C2JRC8 127033410 IC50 = 2800 nM T15334 CYG84R 127033695 IC50 = 10700 nM T15334 C08OEX 127033699 IC50 = 7300 nM T15334 CO8N9D 127033700 IC50 = 3100 nM T15334 C2XM0W 127034291 IC50 = 13900 nM T15334 C34HDE 127048510 IC50 = 325 nM T15334 CWC13T 127048511 IC50 > 10000 nM T15334 CNMU63 127048512 IC50 = 3273 nM T15334 C4HM8S 127048513 IC50 = 716 nM T15334 CHN63B 127048562 IC50 > 10000 nM T15334 C47AMY 127048897 IC50 > 10000 nM T15334 CC63WU 127048898 IC50 > 10000 nM T15334 C0TQH4 127049872 IC50 > 10000 nM T15334 CQ3Z0K 127050169 IC50 > 10000 nM T15334 CQS83M 127050183 IC50 > 10000 nM T15334 C24EST 127050436 IC50 = 84 nM T15334 CGV90M 127050437 IC50 = 3827 nM T15334 C9BRQ1 127050808 IC50 = 60 nM T15334 CKW4P1 127051067 IC50 > 10000 nM T15334 C5B7KM 127052322 IC50 > 10000 nM T15334 CBR62M 127052624 IC50 > 10000 nM T15334 C1D5WM 127053011 IC50 = 826 nM T15334 CL9GD6 127053012 IC50 = 48000 nM T15334 CU3J7F 134131922 IC50 = 520 nM T15334 CV7I9S 134132448 IC50 = 190 nM T15334 CZ6ED0 134134005 IC50 > 50000 nM T15334 C8YAP7 134134664 IC50 = 370 nM T15334 CQ57TZ 134135024 IC50 = 930 nM T15334 CNYB79 134136356 IC50 = 910 nM T15334 CYFN82 134138667 IC50 = 170 nM T15334 C91OAB 134139452 IC50 = 350 nM T15334 C1CI3F 134140475 IC50 = 360 nM T15334 CHI0K8 134141707 IC50 = 3520 nM T15334 CGO03L 134142130 IC50 = 70 nM T15334 CQ5AM4 134143756 IC50 = 60 nM T15334 CKP5H8 134145995 IC50 = 860 nM T15334 CSPO25 134148219 IC50 = 70 nM T15334 CBG21W 134149984 IC50 > 50000 nM T15334 CCKZ27 134150151 IC50 = 420 nM T15334 C13RPI 134150344 IC50 > 50000 nM T15334 C9D8HU 134150865 IC50 = 220 nM T15334 CZ0G4Y 134151297 IC50 = 20970 nM T15334 C2MO8V 134151757 IC50 = 80 nM T15334 CUET51 134152240 IC50 = 6630 nM T15334 CW0OD7 134154514 IC50 > 50000 nM T15334 C12YZE 134154712 IC50 > 50000 nM T15334 CJX52C 134154931 IC50 = 2070 nM T15334 CJ0PS2 134155676 IC50 = 2760 nM T15334 CEYQ01 134156122 IC50 = 300 nM T15334 C9Q1KH 134157378 IC50 = 1620 nM T15334 CH8UD9 134157480 IC50 > 50000 nM T15334 CA12HJ 137632604 IC50 = 4420 nM T15334 CE42VY 137632916 IC50 > 50000 nM T15334 CP0L2R 137637492 IC50 = 4800 nM T15334 CIA47Z 137642031 IC50 = 280 nM T15334 CX8K0G 137647498 IC50 = 200 nM T15334 CO63FM 137650147 IC50 = 510 nM T15334 C8M6WK 137651079 IC50 > 50000 nM T15334 C8YZ7R 137658511 IC50 > 50000 nM T15334 CDZ36P 137659550 IC50 = 1300 nM T15334 C72MWL 137659763 IC50 > 10000 nM T15334 C7EMB5 137660231 IC50 = 3790 nM T15334 C9OI8Z 145954609 IC50 = 10300 nM T15334 C4A1HZ 145957077 IC50 = 38900 nM T15334 D04VCE 44591717 IC50 = 39 nM T15334 D04WPM 9806102 IC50 = 20 nM T15334 D06ATM 91486 IC50 = 12900 nM T15334 D07LUJ 64945 IC50 = 46600 nM T15334 D0C9FK 44591718 IC50 > 3000 nM T15334 D0J4NQ 9847290 IC50 = 156900 nM T39855 C4P8AI 337816 IC50 > 20000 nM T39855 CB6XE5 631160 IC50 > 20000 nM T39855 CG8Y3N 668632 IC50 > 20000 nM T39855 C5TC3I 775009 IC50 = 4100 nM T39855 C0YV5W 775010 IC50 = 2400 nM T39855 CDRW82 873500 IC50 > 20000 nM T39855 C36LSX 956262 IC50 = 8400 nM T39855 C09ZOA 1548433 IC50 = 2300 nM T39855 COA9N6 3268083 IC50 > 20000 nM T39855 C2ZIN8 5345271 IC50 > 20000 nM T39855 CGU4D7 11544962 IC50 = 3500 nM T39855 C6OV3A 11702125 IC50 = 20000 nM T39855 C49EHM 15999508 IC50 > 20000 nM T39855 C1WIT8 20210634 IC50 = 12000 nM T39855 C51JWU 44388739 IC50 > 20000 nM T39855 C6L4EU 44388742 IC50 > 20000 nM T39855 CV4X7H 44388743 IC50 > 20000 nM T39855 C9P4ZK 44388756 IC50 > 20000 nM T39855 CR75SQ 44388766 IC50 > 20000 nM T39855 C84GOQ 44388770 IC50 > 20000 nM T39855 C4JB1K 44388801 IC50 > 20000 nM T39855 CCT1B9 44388828 IC50 = 680 nM T39855 C7WJS4 44388829 IC50 = 750 nM T39855 CU6FQ7 44388831 IC50 > 20000 nM T39855 C45AKR 44388891 IC50 > 20000 nM T39855 CM21JE 44388917 IC50 > 20000 nM T39855 CH6O7U 56927063 IC50 = 640 nM T39855 C4ZGP1 136132244 IC50 > 20000 nM T39855 C0I9OX 136132245 IC50 > 20000 nM T24823 C2ZB4C 5530 IC50 > 100000 nM T24823 CEQ4V8 2723716 IC50 = 34900 nM T24823 CU6S7O 44607264 IC50 = 26000 nM T24823 C1JEG9 46236753 IC50 = 58300 nM T24823 C1FN3T 46830229 Ki = 38000 nM T24823 C35DLK 51049245 IC50 > 100000 nM T24823 CJP68B 71543365 IC50 = 43400 nM T24823 CSM4W0 71616357 IC50 = 49100 nM T24823 CQ3I9J 71616361 IC50 = 36600 nM T24823 CPG73S 73417116 IC50 = 2300000 nM T24823 CI9Q0G 76281715 IC50 = 60000 nM T24823 C05TJO 76282229 IC50 = 230000 nM T24823 CC5IG0 76282703 IC50 > 540000 nM T24823 CA8YE3 76282705 IC50 = 250000 nM T24823 CQ1SM0 102004295 IC50 = 36600 nM T24823 C10VNP 118536083 IC50 = 74700 nM T24823 CF90SQ 118536088 IC50 = 5700 nM T24823 C9T8ZB 118536101 IC50 = 4300 nM T24823 C72EDN 118536105 IC50 = 34700 nM T24823 C9BUT8 118536122 IC50 = 12600 nM T24823 CY2JZ4 118542609 IC50 = 44000 nM T24823 C41EPX 118913669 IC50 > 100000 nM T24823 CJ5NC9 118913682 IC50 > 100000 nM T24823 C1ENW9 118913743 IC50 = 16600 nM T24823 CQNM60 118918087 IC50 = 16700 nM T24823 CGZ1L3 118931167 IC50 = 12900 nM T24823 CLT4M1 127031655 IC50 = 51000 nM T24823 C0C9WI 127032253 IC50 = 11600 nM T24823 CQT5M1 127034333 IC50 = 14900 nM T24823 COY03I 127034334 IC50 = 4300 nM T24823 C97JVF 145948622 IC50 = 7510 nM T24823 C9XO4M 145948655 IC50 = 13200 nM T24823 CHP2V5 145948690 IC50 > 50000 nM T24823 CLD12N 145949023 IC50 = 23200 nM T24823 C5GM0U 145949030 IC50 > 50000 nM T24823 CR34FK 145950671 IC50 = 1430 nM T24823 CX1P7H 145952331 IC50 > 100000 nM T24823 C0TXG3 145954281 IC50 > 100000 nM T24823 CO5NR3 145955440 IC50 = 44800 nM T24823 C5XT4Z 145956132 IC50 > 100000 nM T24823 CPY71F 145956290 IC50 = 4510 nM T24823 C1JKT0 145959891 IC50 > 100000 nM T30829 D0K8KX 5280343 IC50 = 4230 nM T30829 D03HUX 49792852 IC50 > 10000 nM T30829 D0E3TC 44259 IC50 > 10000 nM T30829 D0O0LS 25141092 IC50 > 10000 nM T30829 D0P1CV 46191454 IC50 > 10000 nM T30829 D0Q9UX 16718576 IC50 = 1065 nM T30829 C8IAR2 5281657 IC50 > 100000 nM T30829 CI68PW 5283685 IC50 > 100000 nM T30829 CXK0S6 5283727 IC50 > 100000 nM T30829 C4G9WR 9547398 IC50 > 100000 nM T30829 C76CUP 9547698 IC50 > 100000 nM T30829 CR8DA1 10024683 IC50 > 100000 nM T30829 CLA93G 10047202 IC50 > 100000 nM T30829 C3LCH5 10047545 IC50 > 100000 nM T30829 C4CP7K 10423452 IC50 = 67800 nM T30829 C7HBP6 10429593 IC50 > 10000 nM T30829 C83QWV 10714343 IC50 = 7720 nM T30829 C8G5WP 11210533 IC50 = 1850 nM T30829 C7YG1N 24759534 IC50 = 8800 nM T30829 C5YW7P 24825755 IC50 = 1664 nM T30829 C4EG8R 24993189 IC50 > 10000 nM T30829 CNG96H 25210579 IC50 > 10000 nM T30829 CU3RF1 45139989 IC50 > 10000 nM T30829 CQGZ06 45139991 IC50 > 10000 nM T30829 C7ON5A 46233287 IC50 > 10000 nM T30829 CF91RS 49843531 IC50 > 10000 nM T30829 CBC62W 50899254 IC50 = 595 nM T30829 C2Y6QS 50938552 IC50 > 10000 nM T30829 C9NYP4 51036677 IC50 > 10000 nM T30829 C4WRY3 51037112 IC50 > 10000 nM T30829 CRI28Z 51037948 IC50 > 10000 nM T30829 CE1ZK6 54759168 IC50 > 10000 nM T30829 C9ZFS1 54764923 IC50 > 100000 nM T30829 CBZ8T4 56657856 IC50 = 336 nM T30829 CYPL60 56675140 IC50 > 10000 nM T30829 CXJ63M 59603829 IC50 = 5900 nM T30829 CQEU96 59603842 IC50 = 2600 nM T30829 CV63UL 67240318 IC50 > 10000 nM T30829 C5DGR9 69036886 IC50 = 10000 nM T30829 CCN01X 71547862 IC50 > 10000 nM T30829 C3UC9H 73891099 IC50 = 520 nM T30829 CV8QX0 76310169 IC50 > 30000 nM T30829 CA5L4W 76324771 IC50 > 30000 nM T30829 C9GO0P 76328313 IC50 = 13600 nM T30829 C39FTZ 76335685 IC50 > 100000 nM T30829 C1HW4B 89735655 IC50 = 17000 nM T30829 CY0UC4 90645194 IC50 > 10000 nM T30829 CY7BI2 118706214 IC50 > 10000 nM T30829 C2AN7T 134611886 IC50 > 100000 nM T30829 CHA4N2 136013680 IC50 > 10 nM T30829 C1YUD0 136219394 IC50 > 10 nM T30829 CIU8W3 136254389 IC50 > 10 nM T30829 C2MD1Q 155513187 IC50 > 10000 nM T30829 D03DZO 11715767 IC50 > 10000 nM T30829 D08HFG 24809764 IC50 > 10000 nM T30829 D09HVH 135566652 IC50 > 10 nM T30829 D0C1DQ 6490494 IC50 = 59800 nM T30829 D0T8NU 16757525 IC50 > 4000 nM T29130 D04VIS 5318517 EC50 > 10000 nM T29130 D0J9ZR 4477 IC50 = 250 nM T29130 D01IGZ 10331844 EC50 = 1900 nM T29130 D0JU5X 400769 IC50 = 2380 nM T29130 D0L4FS 5280961 IC50 = 24800 nM T29130 D0MP0X 16659841 IC50 = 23 nM T29130 D03ARS 72550504 Ki = 10000 nM T29130 D03XAK 4253236 IC50 = 74000 nM T29130 D06RBL 73672447 IC50 = 15000 nM T29130 D08EID 72188643 Ki = 10000 nM T29130 D08ETA 76336555 IC50 = 45000 nM T29130 D09ZCV 73333953 IC50 = 12800 nM T29130 D0EX9O 68075823 IC50 = 2800 nM T29130 D0TU0X 252682 Ki = 80000 nM T29130 D0U7LL 53388144 IC50 = 6800 nM T29130 D0V3PA 72545832 Ki = 10000 nM T29130 D0XQ3F 9870708 IC50 = 310000 nM T29130 D0Y0OQ 24767791 Ki = 15000 nM T29130 CZ81DN 87691 IC50 = 14000 nM T29130 CC8QV4 124072 IC50 > 50000 nM T29130 C5X1YU 160254 IC50 = 4600 nM T29130 CS8RE2 160512 IC50 = 14210 nM T29130 C0UL2O 161036 IC50 = 89500 nM T29130 C2BIJ6 442343 IC50 = 73000 nM T29130 CI2KV3 637858 IC50 = 7000 nM T29130 C8U1AQ 658668 IC50 = 20700 nM T29130 CV01HZ 665421 IC50 = 26800 nM T29130 C5C9AV 665426 IC50 = 27000 nM T29130 CX17KE 665524 IC50 > 50000 nM T29130 CYR0A9 665706 IC50 = 21200 nM T29130 C07LUC 665766 IC50 > 50000 nM T29130 CG69BA 665910 IC50 = 6800 nM T29130 C4DWB2 782743 IC50 = 106000 nM T29130 C3K0TB 979808 IC50 = 24320 nM T29130 C1YWC0 987601 IC50 = 60000 nM T29130 C62VHA 1304670 IC50 = 63000 nM T29130 C6RF8N 1334501 IC50 = 144000 nM T29130 CE6JB5 1383290 IC50 = 3700 nM T29130 CSQ26L 1400670 IC50 = 9600 nM T29130 CZJN05 1409627 IC50 = 17900 nM T29130 C4EZ0H 1652812 IC50 = 20000 nM T29130 CBK8I9 1807373 IC50 = 26680 nM T29130 CW3EG8 2104460 IC50 = 75000 nM T29130 C1UVP6 2215480 IC50 = 59910 nM T29130 C3QS1J 2256251 IC50 = 18000 nM T29130 C2XN5M 2779853 IC50 = 5100 nM T29130 CC21YG 3555371 IC50 = 4500 nM T29130 CK27XL 3592521 IC50 = 31200 nM T29130 CJ57WQ 4188928 IC50 = 66000 nM T29130 CFVW35 4219219 IC50 = 61000 nM T29130 CX5JM8 4253237 IC50 = 63000 nM T29130 CLE8J0 4378002 IC50 = 15700 nM T29130 C7IGH6 4655679 IC50 = 3567 nM T29130 CL1A9Z 4744091 IC50 = 7900 nM T29130 CGO70L 5337997 EC50 = 3000 nM T29130 CYT5B9 5340548 IC50 = 91000 nM T29130 C6HKG8 7314631 Ki = 1180 nM T29130 CGJL02 7314633 Ki = 3920 nM T29130 CT0Z1R 9510845 Ki = 1400 nM T29130 C9CTE2 9510848 Ki = 740 nM T29130 C0UVX1 9510856 Ki = 1010 nM T29130 CPL27R 9510868 Ki = 8870 nM T29130 CORG34 9566174 IC50 = 180000 nM T29130 CM10UW 10002209 IC50 = 2200 nM T29130 C5HGS1 10548420 IC50 = 22900 nM T29130 COV54C 10553752 IC50 = 25740 nM T29130 CRKC63 10601247 IC50 > 25000 nM T29130 CA41EF 10673649 IC50 > 25000 nM T29130 C05NWT 10695622 IC50 > 25000 nM T29130 C2L3GK 10719972 IC50 > 25000 nM T29130 CTAP81 10743719 IC50 > 25000 nM T29130 CRF19I 10840295 IC50 > 25000 nM T29130 C7BG3Z 10895852 IC50 = 280 nM T29130 C5QH0J 11228693 IC50 = 6900 nM T29130 CL8BE0 11505560 IC50 = 1400 nM T29130 C2G1PW 11505920 IC50 = 801 nM T29130 C80OQI 11520319 IC50 = 1850 nM T29130 C3WQ8R 11527533 IC50 = 882 nM T29130 CU89MW 11527845 IC50 = 18100 nM T29130 CXT2P8 11541933 IC50 = 748 nM T29130 C0O7KT 11556346 IC50 = 3020 nM T29130 CTLG23 11556428 IC50 = 9810 nM T29130 C04OVM 11578573 IC50 = 596 nM T29130 CQ61YU 11585950 IC50 = 125 nM T29130 C8ZI1W 11607224 IC50 = 2110 nM T29130 C7N1LI 11614102 IC50 = 1780 nM T29130 C34JID 11628749 IC50 = 11800 nM T29130 C8YQ0A 11650282 IC50 = 9780 nM T29130 CF9ZG0 11657425 IC50 = 36600 nM T29130 C3IR9P 11657710 IC50 = 7000 nM T29130 CRDN95 11679384 IC50 = 80000 nM T29130 CFN5G3 11686242 IC50 = 4220 nM T29130 COX46S 11693012 IC50 = 1690 nM T29130 C7OFM8 11700543 IC50 = 1220 nM T29130 C3IP5H 11721811 IC50 = 409 nM T29130 CW5G1P 12967780 IC50 > 25000 nM T29130 CJ3EU2 13245418 IC50 > 50000 nM T29130 C5FH7D 13454179 IC50 = 2500 nM T29130 C36SRY 14586904 IC50 > 50000 nM T29130 CKCD63 15863790 IC50 > 25000 nM T29130 C5U3GA 15944763 IC50 = 3000 nM T29130 C3G5NB 16659060 IC50 = 379 nM T29130 CN89IB 16730520 IC50 = 31000 nM T29130 C6F5HJ 21593530 IC50 = 7000 nM T29130 C9RG3L 24768129 IC50 = 856 nM T29130 CO5QV7 24768157 IC50 > 150000 nM T29130 CZ73XL 24768159 IC50 = 6000 nM T29130 C79KAX 24768160 IC50 = 60000 nM T29130 CLD39N 24768168 IC50 = 6000 nM T29130 C7JT3I 24768169 IC50 = 8000 nM T29130 CP28EL 24768184 IC50 = 620000 nM T29130 CI28CQ 24768185 IC50 = 58000 nM T29130 C37AZQ 24768186 IC50 = 310000 nM T29130 CB5RJ6 24768187 IC50 = 800000 nM T29130 C2B5CI 24768188 IC50 = 58000 nM T29130 CXBZ69 24768189 IC50 = 123000 nM T29130 C1D4AE 24785411 IC50 > 300000 nM T29130 C8WOX3 24785681 IC50 = 86000 nM T29130 CKL1T2 24905706 EC50 = 200 nM T29130 CI2ES6 24905707 EC50 = 170 nM T29130 CVU4B9 24905708 EC50 = 130 nM T29130 C82JKV 25218825 Ki = 350 nM T29130 C0V1ZY 25218826 Ki = 3130 nM T29130 CDI06X 25218827 Ki = 190 nM T29130 CGKU32 42625189 IC50 = 141 nM T29130 C5UZ6L 42625190 IC50 = 233 nM T29130 CK4T0Z 42625191 IC50 = 305 nM T29130 CR3I1V 42625192 IC50 = 25060 nM T29130 CNX56E 42625273 IC50 = 7600 nM T29130 C8HIF3 42625274 IC50 = 7030 nM T29130 CH4GT7 42625275 IC50 = 59800 nM T29130 CCBR08 42625276 IC50 = 195 nM T29130 CVG6F0 42625360 IC50 = 815 nM T29130 C7T8KG 42625361 IC50 = 359 nM T29130 CK10PA 42625362 IC50 = 269 nM T29130 C9PSU4 42625363 IC50 = 35600 nM T29130 CGL2J3 42626364 IC50 = 604 nM T29130 C6GT7R 42626365 IC50 = 45700 nM T29130 CEQZ34 42626366 IC50 = 162 nM T29130 CKE63D 42626367 IC50 = 595 nM T29130 CH70IL 44371812 IC50 = 800 nM T29130 CHR3O5 44371813 IC50 > 6000 nM T29130 CUWO71 44371965 IC50 = 6000 nM T29130 CC2BX6 44371978 IC50 > 6000 nM T29130 CH42RG 44371979 IC50 = 400 nM T29130 CU4IT2 44372037 IC50 = 4000 nM T29130 C2T6YI 44372049 IC50 > 6000 nM T29130 CP16QG 44372105 IC50 = 80000 nM T29130 CD7XO4 44372124 IC50 = 600 nM T29130 C38HPF 44372125 IC50 = 2000 nM T29130 CY7RQ3 44372208 IC50 = 1000 nM T29130 C6B9HZ 44372269 IC50 = 8000 nM T29130 COZ3T6 44372270 IC50 > 6000 nM T29130 CW8F0T 44372304 IC50 = 1600 nM T29130 CI0L6H 44372314 IC50 > 6000 nM T29130 C4GF0M 44372323 IC50 > 6000 nM T29130 CFC98G 44372353 IC50 = 8000 nM T29130 CE3Z8V 44372354 IC50 = 150000 nM T29130 CX3L8P 44372355 IC50 = 30000 nM T29130 CNE92Y 44372391 IC50 = 1000 nM T29130 CEC0Y2 44372543 IC50 = 400 nM T29130 CI0NR5 44372544 IC50 = 1500 nM T29130 CY84EK 44393882 EC50 = 2600 nM T29130 C1L3TA 44404157 IC50 > 100000 nM T29130 CP24SR 44404158 IC50 > 100000 nM T29130 C61BEI 44404159 IC50 > 100000 nM T29130 C6UP3L 44404160 IC50 = 1870 nM T29130 C1SXU6 44404161 IC50 = 484 nM T29130 C8R7SD 44404162 IC50 = 265 nM T29130 CK28NL 44404163 IC50 = 1660 nM T29130 CFT63Q 44404164 IC50 = 1240 nM T29130 C30WHD 44404165 IC50 = 33100 nM T29130 CUHO52 44404166 IC50 = 34600 nM T29130 CC5KM7 44404167 IC50 = 57100 nM T29130 C4D0NZ 44404170 IC50 = 13400 nM T29130 CQ2E9M 44404171 IC50 = 9870 nM T29130 C13LXJ 44404172 IC50 = 13900 nM T29130 C1E3YG 44404803 IC50 = 739 nM T29130 CN72EM 44404804 IC50 = 814 nM T29130 C5FNM7 44404805 IC50 = 497 nM T29130 C9OHC1 44404806 IC50 = 750 nM T29130 C46TJG 44404807 IC50 = 276 nM T29130 COJ53L 44404814 IC50 = 1540 nM T29130 CMCR71 44404815 IC50 = 1070 nM T29130 C39ZDG 44404816 IC50 = 1890 nM T29130 CQ9UD7 44404817 IC50 = 910 nM T29130 C78XFW 44404818 IC50 = 717 nM T29130 C97WEQ 44425197 IC50 = 135 nM T29130 CET6Q3 44425198 IC50 = 850 nM T29130 CR5MI0 44432281 IC50 = 9000 nM T29130 CB03RI 44432282 IC50 = 138000 nM T29130 C5P7EY 44432283 IC50 > 800 nM T29130 C7AC2B 44432285 IC50 > 1000 nM T29130 CD0P1Y 44432286 IC50 > 1000 nM T29130 CBGF73 44432287 IC50 = 108 nM T29130 C28KGO 44473520 IC50 = 110 nM T29130 CRL10C 44473521 IC50 = 1180 nM T29130 CKM3U2 44473522 IC50 = 1880 nM T29130 CYD9A8 44473523 IC50 = 4900 nM T29130 CYEL79 44473524 IC50 = 1350 nM T29130 CZXS83 44473677 IC50 = 848 nM T29130 CAGX43 44473678 IC50 = 294 nM T29130 CW6B9L 44473679 IC50 = 272 nM T29130 CYU8N4 44473680 IC50 = 615 nM T29130 C6U9HV 44473833 IC50 = 1210 nM T29130 CCY43D 44473834 IC50 = 1310 nM T29130 C5H1AI 44473835 IC50 = 1530 nM T29130 C8BS7X 44473836 IC50 = 1080 nM T29130 CD94VT 44473993 IC50 = 1240 nM T29130 C6S4WA 44473994 IC50 = 589 nM T29130 CO20AB 44473995 IC50 = 360 nM T29130 CD4IV3 44473996 IC50 = 797 nM T29130 CU97LI 44473997 IC50 = 454 nM T29130 CS2DJ8 44474160 IC50 = 6900 nM T29130 CF4I5N 44474161 IC50 = 131 nM T29130 CX4B1C 44474162 IC50 = 1350 nM T29130 C8L2CT 44474163 IC50 = 68 nM T29130 C0XL2F 44474307 IC50 = 303 nM T29130 CW3EO9 44474308 IC50 = 175 nM T29130 CYEH20 44474309 IC50 = 1630 nM T29130 CHIJ36 44474310 IC50 = 437 nM T29130 CU90IR 44474458 IC50 = 94 nM T29130 CAC61N 44474949 IC50 = 511 nM T29130 CP0CA2 44474950 IC50 = 499 nM T29130 C1F2XP 44475086 IC50 = 69 nM T29130 C3ZLC0 44475230 IC50 = 290 nM T29130 CIDZ45 44475556 IC50 = 4940 nM T29130 CL9YQ6 44475557 IC50 = 874 nM T29130 C8LE3Z 44475558 IC50 = 1400 nM T29130 C4MXS0 44475559 IC50 = 11400 nM T29130 CNHU20 44475710 IC50 = 574 nM T29130 CSL74Q 44475712 IC50 = 1140 nM T29130 C5CIX9 44475713 IC50 = 3310 nM T29130 CS8NP7 44475714 IC50 = 3210 nM T29130 CC04JX 44475868 IC50 = 7800 nM T29130 CD6KB7 44475869 IC50 = 3600 nM T29130 C0D9LJ 44475870 IC50 = 68200 nM T29130 CK5IS1 44475871 IC50 = 2640 nM T29130 CB2Y1Q 44475872 IC50 = 1830 nM T29130 C5GCO6 44568723 EC50 = 4600 nM T29130 CIEM82 44568724 EC50 = 46000 nM T29130 CA0ZQ6 44580433 IC50 = 357000 nM T29130 CH4WU1 44582627 IC50 = 231 nM T29130 C4L3ZT 44582628 IC50 = 150 nM T29130 CO4R8Y 44582630 IC50 = 136 nM T29130 CCEJ32 44582631 IC50 = 186 nM T29130 C7MC1D 44582632 IC50 > 100000 nM T29130 C0MA7J 44582633 IC50 > 100000 nM T29130 CL4Q2P 44582635 IC50 > 100000 nM T29130 CA8NP0 44582636 IC50 = 3530 nM T29130 CI53ZJ 44582637 IC50 = 24700 nM T29130 CVH18D 44582638 IC50 = 1650 nM T29130 C3S5ZU 44582639 IC50 = 4640 nM T29130 CY3DS8 44582640 IC50 = 3240 nM T29130 CFWU57 44582641 IC50 = 190 nM T29130 CT5FW6 44582682 IC50 = 19200 nM T29130 C1HO9G 44583885 IC50 = 15840 nM T29130 C9IF7E 45105600 Ki = 2500 nM T29130 C4NI8L 45483580 IC50 = 69 nM T29130 CJ8U5F 45483592 IC50 = 1110 nM T29130 C14KEZ 46938290 Ki = 18700 nM T29130 C0F4ZU 49779985 EC50 = 15000 nM T29130 C9L3XR 49838879 IC50 > 10000 nM T29130 CU6VH8 49862810 IC50 = 24800 nM T29130 C14EZS 53247983 Ki = 66 nM T29130 C9B2QA 53247984 Ki = 43 nM T29130 CSV3O4 53247985 Ki = 48 nM T29130 CD4SO8 53247986 Ki = 33 nM T29130 C4V3BF 53248037 Ki = 57 nM T29130 CO3XT2 53248554 Ki = 144 nM T29130 CY20XT 53248591 Ki = 203 nM T29130 C74ERM 53248592 Ki = 94 nM T29130 CPM1G0 53248593 Ki = 83 nM T29130 C2PU8L 53248594 Ki = 193 nM T29130 C8LUY0 53248595 Ki = 39 nM T29130 CGW5S7 53248606 Ki = 386 nM T29130 C0RF7E 53248629 Ki = 66 nM T29130 CLD5E3 53248630 Ki = 114 nM T29130 C5IR2F 53248631 Ki = 46 nM T29130 CEK5T9 53248632 Ki = 105 nM T29130 C36AOD 53248633 Ki = 188 nM T29130 C9MU3N 53249071 IC50 > 50000 nM T29130 C0ACV7 53318421 IC50 = 55000 nM T29130 CN9OM4 53319752 IC50 = 72000 nM T29130 C2DVZ6 53321048 IC50 = 66000 nM T29130 CNP8C1 53323751 IC50 = 75000 nM T29130 C0U7KR 53325584 IC50 = 34540 nM T29130 CJG32W 56659993 Ki = 26500 nM T29130 CF15NC 56663448 Ki = 8000 nM T29130 CXU2Q3 56663449 Ki > 100000 nM T29130 C9LP8R 56663450 Ki = 30600 nM T29130 CZI54O 56673821 Ki = 11000 nM T29130 CO7R8N 56680467 Ki = 6200 nM T29130 C2WDB7 56680468 Ki = 13300 nM T29130 C2MX8E 56683798 Ki = 41000 nM T29130 C0HSI2 56847442 Ki = 8400 nM T29130 CD1V5I 56847565 IC50 = 14400 nM T29130 CY59KF 56847566 IC50 = 14400 nM T29130 CM3TY5 56847620 IC50 = 22000 nM T29130 CW6KE5 57380393 IC50 = 110000 nM T29130 C3X2FY 57384017 IC50 = 6300 nM T29130 C2HPR0 57395002 EC50 = 5050 nM T29130 CDO01I 57396749 EC50 = 1180 nM T29130 CHG58S 68075821 IC50 = 6200 nM T29130 CZ2KU9 68075824 IC50 = 5000 nM T29130 C64MBD 68075825 IC50 = 46600 nM T29130 CPF83Q 68075827 IC50 = 12400 nM T29130 CKU2G7 68075828 IC50 = 22600 nM T29130 CLQ8U6 68075829 IC50 = 7600 nM T29130 C76RSC 68075831 IC50 = 9000 nM T29130 CO2Q8P 68075832 IC50 > 50000 nM T29130 CQ49AV 68075834 IC50 = 7200 nM T29130 C5XHR8 68075842 IC50 = 9200 nM T29130 C2IXG3 68075843 IC50 = 10600 nM T29130 CA67TH 68075844 IC50 = 9600 nM T29130 CN36CH 68075846 IC50 = 11000 nM T29130 CSL3N8 68075861 Ki = 2800 nM T29130 CU9EB8 68075862 IC50 > 50000 nM T29130 C1P2HG 68075866 IC50 = 15800 nM T29130 CJP40C 68075867 IC50 = 8800 nM T29130 C1PSI4 68075868 IC50 = 11800 nM T29130 CYLB93 68075871 IC50 > 300000 nM T29130 CO5WQ1 68075872 IC50 = 11000 nM T29130 CN9J6D 68075873 IC50 = 17800 nM T29130 CQYA27 68075874 IC50 = 12400 nM T29130 CN8F6G 68075880 IC50 = 7600 nM T29130 CH7V3Q 68075882 IC50 = 10200 nM T29130 CG4X3J 68075885 IC50 > 50000 nM T29130 C93ZOA 68075889 IC50 = 45200 nM T29130 C3G6TY 68075890 IC50 = 11600 nM T29130 C26MPF 68075895 IC50 = 5000 nM T29130 C0UMX5 68075897 IC50 = 6000 nM T29130 C4HZJ3 68075906 IC50 = 5200 nM T29130 COFR74 68075908 IC50 = 18400 nM T29130 CSN9P1 68075975 IC50 = 8000 nM T29130 CU61YT 68075994 Ki = 7900 nM T29130 C9L4PU 68076002 IC50 > 50000 nM T29130 CQ5WT2 68076014 IC50 = 24000 nM T29130 CL64DJ 68076215 IC50 = 8600 nM T29130 CCTW23 68076216 IC50 = 14400 nM T29130 C70SUO 68076254 IC50 = 17000 nM T29130 CH7NC1 68076255 IC50 = 10000 nM T29130 CAYX80 68076759 Ki > 25000 nM T29130 C9SMV3 68815772 IC50 = 35700 nM T29130 CT2G3X 70681428 Ki = 8400 nM T29130 C1VM0Q 70681429 Ki = 17600 nM T29130 CKHZ34 70692803 IC50 = 3200 nM T29130 C2C5ID 71449913 IC50 = 43000 nM T29130 CJW1B8 71451245 IC50 = 32500 nM T29130 C7R5EZ 71571581 IC50 = 15600 nM T29130 C6UG1V 71653594 IC50 = 1600 nM T29130 CUM45G 71680713 Ki = 2500 nM T29130 C6Z8PV 71725229 IC50 > 50000 nM T29130 CL34JM 71726961 Ki = 13300 nM T29130 CB74ON 71812276 Ki = 18200 nM T29130 C8JC0Z 72374404 IC50 = 11000 nM T29130 C4I3ZY 73333711 IC50 = 20800 nM T29130 C15GQP 73333832 IC50 = 32400 nM T29130 CEZ57I 73333833 IC50 = 20600 nM T29130 C3V8KZ 73333834 IC50 = 27400 nM T29130 CIX7C5 73333951 IC50 = 11800 nM T29130 CIU35L 73333952 IC50 = 14600 nM T29130 CI3X5T 73333954 IC50 = 9600 nM T29130 C1F7HM 73334053 IC50 = 28000 nM T29130 C2C6SF 73334054 IC50 = 17800 nM T29130 CMT46F 73334055 IC50 = 17600 nM T29130 CLN46T 73334056 IC50 = 11000 nM T29130 C73MCN 73334149 IC50 = 18200 nM T29130 C9J5RZ 73334150 IC50 = 13800 nM T29130 CZKO45 73334151 IC50 = 10200 nM T29130 C36QFL 73334152 IC50 = 17800 nM T29130 C45YCM 73334248 IC50 = 21600 nM T29130 CL93GF 73334249 IC50 = 11400 nM T29130 CV5NZ0 73334250 IC50 = 19800 nM T29130 CKJV17 73334251 IC50 = 9400 nM T29130 COM2J6 73334350 IC50 = 12400 nM T29130 CT51JG 73334351 IC50 = 17600 nM T29130 C60POI 73334352 IC50 = 16600 nM T29130 C8M7QV 73334463 IC50 = 21800 nM T29130 C27GIZ 73334464 IC50 = 17400 nM T29130 CI9F7O 73334576 IC50 = 30800 nM T29130 CAKM84 73334678 IC50 = 22200 nM T29130 C69GVQ 73334679 IC50 = 15400 nM T29130 CLBC87 73334680 IC50 = 22800 nM T29130 C1TX5V 73334681 IC50 = 8100 nM T29130 C41KAC 73345548 IC50 = 20000 nM T29130 C82TQB 73345635 Ki = 7300 nM T29130 CV1A6H 73345657 IC50 > 100000 nM T29130 C9M2TL 73346330 IC50 > 300000 nM T29130 CV3YI8 73346331 IC50 = 95000 nM T29130 C5XO2M 73348950 IC50 > 50000 nM T29130 C5OUL0 73352819 IC50 = 300 nM T29130 C9CJ0U 73353126 IC50 > 150000 nM T29130 C7INR4 73356550 IC50 = 22400 nM T29130 CG46NZ 74221732 IC50 = 42000 nM T29130 C74PLG 74221733 IC50 = 28400 nM T29130 C3UVG1 74221822 IC50 = 118100 nM T29130 CYK38B 74221824 IC50 = 48000 nM T29130 C29SMB 74221912 IC50 = 52000 nM T29130 C0R5OB 74221913 IC50 = 12800 nM T29130 C28UPN 74221914 IC50 = 32000 nM T29130 CRWE15 74221915 IC50 = 33300 nM T29130 C2JEN9 76311218 IC50 = 22000 nM T29130 C5RCX8 76311219 IC50 = 43000 nM T29130 C1S7GV 76311220 IC50 = 22200 nM T29130 C9DGQ0 76314830 IC50 = 22000 nM T29130 C6R8YS 76318440 IC50 = 20000 nM T29130 C03URV 76322104 IC50 = 18900 nM T29130 CAM9C7 76322107 IC50 > 1000000 nM T29130 CY6J1N 76322108 IC50 = 57000 nM T29130 C9YG8K 76325718 IC50 > 300000 nM T29130 C47AHC 76325719 IC50 = 33500 nM T29130 CYQG59 76325720 IC50 = 50000 nM T29130 COVY87 76325721 IC50 = 23300 nM T29130 CCW94L 76325722 IC50 = 19000 nM T29130 C0BR6K 76325723 IC50 = 17000 nM T29130 C1NYJ6 76329292 IC50 = 23000 nM T29130 CD06NW 76332943 IC50 = 50000 nM T29130 C01UMA 76332944 IC50 = 35300 nM T29130 CXK4A5 76332945 IC50 = 15000 nM T29130 C5SZ6G 76332946 IC50 = 61000 nM T29130 CFD52M 76332947 IC50 = 32000 nM T29130 C43UEN 76336554 IC50 = 94700 nM T29130 C49ZYI 76336556 IC50 = 201300 nM T29130 C5YA0B 81689912 IC50 = 2400 nM T29130 C8G2OH 86581489 IC50 = 500 nM T29130 C0EX1K 86581491 IC50 = 500 nM T29130 CMZI69 86581492 IC50 = 500 nM T29130 CS1UO7 86581493 IC50 = 500 nM T29130 COZ06A 86581639 IC50 = 500 nM T29130 CU6E0X 90644814 IC50 = 19400 nM T29130 CD4IR5 90665637 IC50 = 17700 nM T29130 C9SY6A 101805555 IC50 = 590 nM T29130 C8SB0X 101805556 IC50 = 17100 nM T29130 C6Z9TW 102004285 Ki = 143800 nM T29130 C49FBG 118318714 Ki = 440 nM T29130 C34BNA 118714785 IC50 > 30000 nM T29130 CSMF46 118714786 IC50 > 30000 nM T29130 C5MXD3 118714787 IC50 > 30000 nM T29130 C1L6DR 118714788 IC50 > 30000 nM T29130 CXAK53 118714789 IC50 > 30000 nM T29130 CO4ZX1 118714790 IC50 > 30000 nM T29130 C80IVZ 118714791 IC50 > 30000 nM T29130 C1Z8UW 118714792 IC50 > 30000 nM T29130 CS4Y6R 118714793 IC50 > 30000 nM T29130 CGO49H 121485603 IC50 = 8200 nM T29130 CKZB63 122179017 IC50 > 30000 nM T29130 C68DWU 122179018 IC50 > 30000 nM T29130 C3QD5E 122179019 IC50 > 30000 nM T29130 CJ98AX 122179020 IC50 > 30000 nM T29130 C3TM6O 122179021 IC50 = 19200 nM T29130 CS2F3X 122179022 IC50 = 270 nM T29130 CDX76J 122179023 IC50 = 17600 nM T29130 C39GEA 122179024 IC50 = 4000 nM T29130 C6TJ1C 122179025 IC50 = 500 nM T29130 C4B8MR 122184505 IC50 = 4020 nM T29130 CTL07X 122184507 IC50 = 440 nM T29130 C4P5KU 122184516 IC50 = 2750 nM T29130 C7WSP6 122184518 IC50 = 200 nM T29130 C3AI9V 122184592 IC50 = 320 nM T29130 CU3V7O 122193685 IC50 = 25700 nM T29130 C0FY5O 122195118 IC50 = 610000 nM T29130 CQD86F 122417980 IC50 = 9100 nM T29130 CZ6C3I 124585685 IC50 = 67000 nM T29130 CWP4Y3 127043537 IC50 > 50000 nM T29130 CD4PS6 127043538 IC50 > 30000 nM T29130 C3Z6WV 127043646 IC50 = 15500 nM T29130 C62JRB 127043708 IC50 > 50000 nM T29130 CYK0A6 127043709 IC50 > 50000 nM T29130 CZ2J7S 127043710 IC50 > 50000 nM T29130 CRMT13 127043884 IC50 > 50000 nM T29130 CVQR69 127043885 IC50 = 11000 nM T29130 CWT75I 127043886 IC50 > 50000 nM T29130 CBPX56 127043998 IC50 = 5600 nM T29130 C5J8LF 127044001 IC50 > 50000 nM T29130 CDO20J 127044052 IC50 > 50000 nM T29130 CN27VG 127044282 IC50 = 2200 nM T29130 CNJ8A1 127044345 IC50 = 21200 nM T29130 CWM68F 127044476 IC50 = 5100 nM T29130 C65KPY 127044624 IC50 = 4200 nM T29130 CA6WV5 127044625 IC50 = 5720 nM T29130 CIXY97 127044626 IC50 = 4400 nM T29130 C7MIB0 127044627 IC50 = 4100 nM T29130 CP0KI6 127044628 IC50 = 7500 nM T29130 C9BJ7M 127044629 IC50 > 20000 nM T29130 CV79XP 127044630 IC50 > 50000 nM T29130 CJ5SF0 127044631 IC50 = 18600 nM T29130 CYH75N 127044796 IC50 = 7500 nM T29130 C4PV9O 127044955 IC50 = 3400 nM T29130 CF3IT2 127045104 IC50 = 3800 nM T29130 CF62PM 127045575 IC50 = 14500 nM T29130 C7E5CW 132583591 IC50 > 50000 nM T29130 CRG46C 134134277 IC50 = 38660 nM T29130 CAT0S5 134135330 IC50 > 50000 nM T29130 CHN5U8 134136919 IC50 > 50000 nM T29130 CUXZ40 134143020 IC50 > 50000 nM T29130 CFC40X 134146883 IC50 > 50000 nM T29130 C7U4LT 134152352 IC50 > 50000 nM T29130 CO6SK5 134155047 IC50 > 50000 nM T29130 CK78JZ 134157370 IC50 > 50000 nM T29130 C1QXI7 135402276 IC50 = 6400 nM T29130 CBN8M7 135449231 IC50 = 5000 nM T29130 CJ58AO 135463175 IC50 = 33900 nM T29130 CSB0M9 135494223 IC50 = 16200 nM T29130 CX4ZB3 135863110 IC50 = 1700 nM T29130 CST9B8 136244569 IC50 = 18200 nM T29130 CSK95Y 136504263 IC50 > 50000 nM T29130 CW6YH7 139600322 Ki = 14 nM T29130 CU7VO6 141744834 IC50 = 640 nM T29130 CYKD76 141744836 IC50 = 990 nM T29130 CG7PH4 145949574 IC50 = 11900 nM T29130 C2A5NK 145949658 EC50 = 3450 nM T29130 C2B8HT 145950270 EC50 = 2230 nM T29130 CF85PT 145950476 EC50 > 10000 nM T29130 C7VWP9 145950692 EC50 = 800 nM T29130 C2J3NX 145950701 EC50 = 4160 nM T29130 CXCE08 145951232 EC50 = 3950 nM T29130 CJZ26R 145951538 EC50 = 8180 nM T29130 C81CPI 145951661 IC50 = 52600 nM T29130 C5TX9Z 145951774 IC50 = 47000 nM T29130 C65WDU 145952038 IC50 = 43000 nM T29130 CB5G6C 145952840 IC50 > 100000 nM T29130 C78DHC 145953545 EC50 > 10000 nM T29130 C46LXG 145953816 IC50 = 71900 nM T29130 C6JF8R 145954862 EC50 = 5380 nM T29130 C1F3AC 145955014 EC50 = 3050 nM T29130 CYEM89 145955153 EC50 = 4400 nM T29130 C3ZM6K 145955473 EC50 > 10000 nM T29130 C56ATB 145955610 EC50 > 10000 nM T29130 C25NVA 145956182 IC50 = 27600 nM T29130 CSY98I 145956215 EC50 = 990 nM T29130 CP7KH1 145956218 IC50 > 100000 nM T29130 CN61YR 145956444 EC50 > 10000 nM T29130 CFS34O 145956557 IC50 = 40500 nM T29130 CY2A3C 145956686 IC50 = 29700 nM T29130 CP41CN 145957009 EC50 > 10000 nM T29130 CI64ZE 145957487 EC50 = 3110 nM T29130 CC1SP5 145957565 IC50 = 79100 nM T29130 CRC2T0 145957761 EC50 = 2550 nM T29130 C89VLM 145957890 EC50 = 6100 nM T29130 CIV05T 145958301 EC50 = 4750 nM T29130 C8WT3G 145958620 EC50 = 5380 nM T29130 C9OH8Y 145958729 EC50 = 4340 nM T29130 CRE9K0 145958784 EC50 = 3220 nM T29130 CD5U1R 145958841 IC50 = 12200 nM T29130 CFM3D1 145959802 IC50 = 21900 nM T29130 C76UXC 145960795 EC50 > 10000 nM T29130 CG4A8P 145962477 EC50 = 5680 nM T29130 C8LH6C 145963539 IC50 > 100000 nM T29130 C62RLG 145963983 IC50 > 25000 nM T29130 C2QVC5 145964968 IC50 > 25000 nM T29130 COGN67 145965850 IC50 > 25000 nM T29130 CTCE64 145965867 IC50 > 25000 nM T29130 C31UPV 145965989 IC50 > 25000 nM T29130 CI6CL4 145966660 IC50 > 25000 nM T29130 CQ37MK 145969977 IC50 = 10000 nM T29130 C6JPF5 145972166 EC50 > 10000 nM T29130 C2N8GQ 145972173 IC50 = 19400 nM T29130 CN1CR5 145972237 EC50 = 5810 nM T29130 CGS71T 145972484 IC50 > 100000 nM T29130 CU3C6Q 145973136 EC50 > 10000 nM T29130 C9GF6X 145974814 IC50 > 100000 nM T29130 CP68JQ 145977608 IC50 > 25000 nM T29130 CWK1C6 155188865 Ki = 12 nM T29130 C1Y4WZ 155189019 Ki = 14 nM T29130 C9IM3A 155189022 Ki = 7 nM T29130 C8XUI5 155189027 Ki = 25 nM T29130 C8J0NQ 155189031 Ki = 14 nM T29130 CV3Z5E 155516315 Ki = 33 nM T29130 CNU4S2 155518066 Ki = 21900 nM T29130 C2CER4 155528099 IC50 = 13020 nM T29130 CIMP57 155528643 Ki = 761 nM T29130 C27LIG 155537212 IC50 = 2280 nM T29130 C3PA7Z 155544860 Ki = 584 nM T29130 CC84LS 155549005 Ki = 164 nM T29130 CTG39A 155552041 Ki = 7300 nM T29130 CK3FU1 155552413 IC50 = 5070 nM T29130 C6S4QJ 155555870 IC50 = 23980 nM T29130 CD7XV1 155559738 IC50 = 9130 nM T29130 C3FSL6 155567563 IC50 = 15140 nM T29130 CSQ54Y 24768128 IC50 = 739 nM T29130 D0IO0I 6474893 IC50 = 6000 nM T29130 D0JW1C 53386731 IC50 > 50000 nM T29130 D0SJ2Q 10494 IC50 > 50000 nM T64567 D00STL 644241 Ki = 41.9 nM T64567 D00ZOF 23666456 Ki > 150000000 nM T64567 D01MUR 68844 Ki = 36 nM T64567 D02FLB 516892 Ki = 13000000 nM T64567 D02PJA 24841 Ki = 7000000 nM T64567 D02URS 4875 Ki = 7000000 nM T64567 D03QGM 5355 Ki = 31 nM T64567 D03RTS 2662 Ki = 16 nM T64567 D03UOT 785 Ki = 32500 nM T64567 D05OFX 219078 Ki = 353 nM T64567 D05UYW 5284549 Ki = 52 nM T64567 D07CWD 3657 Ki = 23000 nM T64567 D07HBX 338 Ki = 78700 nM T64567 D07INV 3295 IC50 = 0.25 nM T64567 D07VDZ 5284627 Ki = 58 nM T64567 D09NIA 2732 Ki = 23 nM T64567 D09VAZ 5565 Ki = 39000 nM T64567 D0AZ3C 5291 Ki = 75.7 nM T64567 D0AZ8C 5213 Ki = 10150 nM T64567 D0C2II 4100 Ki = 27 nM T64567 D0C8EU 5394 Ki > 50000 nM T64567 D0C8FX 3005837 Ki = 1720 nM T64567 D0E1SW 1986 Ki = 0.06 nM T64567 D0E9JM 4873 Ki = 33000000 nM T64567 D0H8FH 3702 Ki = 36 nM T64567 D0J4GO 3038 Ki = 34 nM T64567 D0J7RK 36811 Ki = 9820 nM T64567 D0K0OZ 5702160 Ki = 126.3 nM T64567 D0K1QD 3998 Ki = 103 nM T64567 D0K8KX 5280343 Ki = 7000 nM T64567 D0L4JT 5333 Ki = 238 nM T64567 D0L6DA 119607 IC50 = 27 nM T64567 D0L7FM 4911 Ki = 360 nM T64567 D0OT0O 44561 Ki = 2210000 nM T64567 D0PQ3G 3440 Ki = 420 nM T64567 D0SH3I 387447 Ki = 3380 nM T64567 D0TG1H 3033 IC50 > 100000 nM T64567 D0U5QK 1983 Ki = 70700 nM T64567 D0V8QT 2708 Ki > 50000 nM T64567 D0VM2L 68740 IC50 = 5323 nM T64567 D0W5HK 216239 Ki > 10000 nM T64567 D0Y2IZ 5560 Ki = 87 nM T64567 D0Z3EI 6038 Ki = 82 nM T64567 D0Z4UY 517045 Ki > 150000000 nM T64567 D02ECG 23662274 Ki = 1120000 nM T64567 D04IIU 216468 Ki = 24 nM T64567 D05NJI 5287541 Ki = 34 nM T64567 D05ZXZ 491941 Ki = 81 nM T64567 D06DMQ 59472121 Ki > 50000 nM T64567 D06PII 5356 Ki = 43 nM T64567 D07ZNI 9804302 Ki = 70 nM T64567 D08BXT 1102 Ki = 1370 nM T64567 D09XQU 135413511 Ki > 50000 nM T64567 D0L6HN 996 Ki = 8800 nM T64567 D0SC6I 517055 Ki > 150000000 nM T64567 D0U3EP 445154 Ki = 810 nM T64567 D0V0UK 82267 Ki = 9600 nM T64567 D03SLR 445858 Ki = 9870 nM T64567 D08RPE 71607911 IC50 > 3900 nM T64567 D0F8XZ 19890 Ki = 6700 nM T64567 D0NH9P 135 Ki = 3730 nM T64567 D0X2AU 23427 Ki > 100000 nM T64567 D07XPE 8249 Ki > 50000 nM T64567 D0LD9S 1103 Ki = 13300 nM T64567 CI0WH9 72 Ki = 4450 nM T64567 CUT2V4 260 Ki = 16000000 nM T64567 COV5W3 402 Ki = 7000 nM T64567 CSZ43B 540 Ki = 40000 nM T64567 C97QXH 767 Ki = 8600 nM T64567 C39CTO 768 Ki = 4000 nM T64567 C1QDT0 781 Ki = 130000 nM T64567 CW0R2L 944 Ki = 46000000 nM T64567 C2LNM9 1016 Ki = 1230000 nM T64567 C8W7BZ 1118 Ki = 154000000 nM T64567 CU12QE 1203 Ki = 5030 nM T64567 C6O0MZ 1491 Ki = 68000 nM T64567 CO4X7B 2456 IC50 = 90 nM T64567 C5L7VX 2871 Ki = 6410 nM T64567 CZP5J2 3415 Ki = 2210000 nM T64567 CQ0D8J 3469 Ki = 6600 nM T64567 CJ2F6P 5056 Ki = 9530 nM T64567 CDJ4K6 5987 Ki = 9200 nM T64567 CU9EM3 6125 Ki = 3280000 nM T64567 CUP2F4 7043 Ki = 8630 nM T64567 C1CVT7 7121 Ki = 8250 nM T64567 C6NC4O 7414 Ki = 5640 nM T64567 CJKY76 7420 Ki = 4530 nM T64567 C23KMD 7921 Ki = 920 nM T64567 C6QYD8 8434 Ki = 8200 nM T64567 CXF7C6 8736 Ki = 7420000 nM T64567 CR3IF4 8865 Ki = 1270000 nM T64567 CHP7I1 9016 Ki = 4150 nM T64567 CLYZ50 9338 Ki = 5900 nM T64567 CNM7L3 10199 Ki = 174 nM T64567 CBIR94 10313 Ki = 45900 nM T64567 CC30SK 10341 Ki = 4420 nM T64567 CACI42 10953 Ki = 3660 nM T64567 CV5PC3 11568 Ki = 4900 nM T64567 CL80QG 11820 Ki = 44.6 nM T64567 C14BYX 12662 Ki = 2470 nM T64567 C57OTC 13818 Ki = 1260000 nM T64567 CKA21F 14768 Ki = 2750000 nM T64567 CUA0L6 14917 Ki = 48000000 nM T64567 CNI85U 15109 Ki = 9070 nM T64567 CS8X0P 16124 Ki = 860000 nM T64567 CQ4C5U 16523 Ki = 890 nM T64567 CS39YR 19654 Ki = 147000000 nM T64567 CNGB21 20098 Ki = 910 nM T64567 C3LA1Z 20161 Ki = 7400 nM T64567 CMK0O4 20825 Ki = 223 nM T64567 CF14KR 24247 Ki = 11600000 nM T64567 C4IZB8 24345 Ki = 49700000 nM T64567 C9M8EJ 24434 Ki = 46000000 nM T64567 C8S9AF 24445 Ki = 274000000 nM T64567 CFM9L6 24530 Ki = 5000 nM T64567 CG04AY 26518 Ki > 100000 nM T64567 CDK20Z 27290 Ki = 400 nM T64567 C69RDT 32204 Ki = 4130 nM T64567 C7YZM4 33557 Ki = 5000 nM T64567 C4OU6D 35703 Ki = 9600 nM T64567 CDIJ43 36573 Ki = 2400 nM T64567 C89DPG 39981 Ki = 2250000 nM T64567 CY2GU3 60582 Ki = 12.8 nM T64567 CF26VS 61441 Ki = 35200000 nM T64567 CLMR98 61857 Ki = 3630000 nM T64567 C5MJH8 64789 Ki = 610 nM T64567 CN94KU 65008 Ki = 830 nM T64567 C6DG9Q 65185 Ki = 30300000 nM T64567 C1NQ8E 65188 Ki = 7510 nM T64567 CT6YO0 66548 Ki = 740 nM T64567 CCE63L 66634 IC50 = 588.34 nM T64567 CMXS19 66814 Ki = 26.1 nM T64567 CJ1Z2R 67125 Ki = 15700 nM T64567 C0ZK7U 67284 Ki = 4060 nM T64567 CWXE69 67756 Ki = 116 nM T64567 C26PTJ 67760 Ki = 349 nM T64567 CJWD84 68154 Ki = 1600 nM T64567 CA3R7P 68351 Ki = 34 nM T64567 CX4HM3 70653 IC50 = 217 nM T64567 CI80QC 71485 Ki = 2200 nM T64567 C8U0VH 72597 Ki = 37.5 nM T64567 CU79WI 74093 Ki = 235 nM T64567 CTMF08 75076 Ki = 810 nM T64567 C0I4UT 75077 Ki = 840 nM T64567 C7L1RO 75522 Ki = 6.6 nM T64567 CE5RZ1 76509 Ki = 310 nM T64567 C9V0ME 77547 Ki = 780 nM T64567 C6TS8J 77548 Ki = 860 nM T64567 CRXH06 77553 Ki = 151.8 nM T64567 CX47BZ 78479 Ki = 48000 nM T64567 CCK8E1 79611 Ki = 10.8 nM T64567 CYIP60 89607 Ki = 27 nM T64567 CM72DQ 90631 Ki = 120 nM T64567 CB5R7Y 92229 Ki = 350 nM T64567 CB81UG 93577 Ki = 93 nM T64567 C2GI9X 95801 IC50 = 76 nM T64567 C40RWH 95840 Ki = 140 nM T64567 C21JNS 95841 Ki = 89.2 nM T64567 C1GQE3 97576 Ki = 3100 nM T64567 CA9YN2 99477 Ki = 30.5 nM T64567 CV76MT 100187 Ki = 95.8 nM T64567 CGM6A9 101263 Ki > 1000 nM T64567 C6K3MG 101424 Ki > 100000 nM T64567 CDP5M6 125623 Ki = 143 nM T64567 CN19UT 129695 Ki = 120 nM T64567 CCK5Y6 133125 Ki = 2.7 nM T64567 CVB67D 134560 Ki = 38 nM T64567 CUBQ92 145746 Ki > 1000 nM T64567 C9ZEP5 151399 Ki > 1000 nM T64567 C47BCV 154989 Ki = 1320 nM T64567 CJ0FR9 155148 Ki = 860 nM T64567 C50XVJ 159772 Ki = 2560 nM T64567 CVH81Y 163571 Ki = 30 nM T64567 C8AO0Z 165323 Ki = 30 nM T64567 C6M0TK 167985 Ki = 330000 nM T64567 CU3WG6 179620 Ki = 8120 nM T64567 CE1VJ6 191826 Ki = 3200 nM T64567 CO96LR 192271 Ki = 26 nM T64567 C1N3AY 199210 Ki > 100000 nM T64567 C2GHM7 202375 IC50 = 94 nM T64567 C9K3VU 220023 IC50 = 93 nM T64567 CEZU63 221227 Ki = 2450 nM T64567 C7DS2I 228958 Ki = 13.7 nM T64567 C2ED9N 236541 Ki = 236 nM T64567 C14USE 239728 Ki = 290 nM T64567 CW1E5G 239730 Ki = 290 nM T64567 C6D1LY 246499 Ki = 4.9 nM T64567 C0B3OQ 253877 Ki = 16000000 nM T64567 CLV79E 260228 Ki = 4350 nM T64567 CU45WA 260244 Ki > 100000 nM T64567 C3QV5H 287064 Ki = 790 nM T64567 C26HNY 289493 Ki = 890 nM T64567 C83MLQ 295450 Ki = 230 nM T64567 COE9A7 306924 Ki = 575 nM T64567 CAUO79 306968 Ki = 7.7 nM T64567 CM2N3X 307505 Ki = 8.4 nM T64567 C3W0AQ 307522 Ki = 465 nM T64567 C3WZI1 308397 Ki = 952 nM T64567 C6AKQ8 308411 Ki = 41.5 nM T64567 CL4GF1 308432 Ki = 35.6 nM T64567 C96DKW 310360 Ki = 45 nM T64567 CY13EN 311156 Ki = 7.3 nM T64567 C12PJC 313721 IC50 = 128 nM T64567 COI7H8 317746 Ki = 3.9 nM T64567 CG3J6Q 323350 Ki = 4.1 nM T64567 CTX0Z3 327169 Ki = 730 nM T64567 CXZ14S 341082 Ki > 50000 nM T64567 CP7X9H 342056 Ki = 30.1 nM T64567 CMS5W4 343662 Ki = 164 nM T64567 CH1C9B 351361 Ki = 506 nM T64567 CM9V8O 388547 Ki = 18 nM T64567 CT3ZU4 388776 Ki = 11400 nM T64567 CH21KA 389641 Ki = 124000 nM T64567 C6CQO3 389642 Ki = 144000 nM T64567 CH0F9P 390929 Ki = 210 nM T64567 CNPZ40 394897 Ki = 6.4 nM T64567 CHU17A 395815 Ki = 75 nM T64567 CA8C5N 439514 Ki = 8720 nM T64567 CC54LQ 450256 IC50 = 8922 nM T64567 C5IPL1 471796 Ki = 724 nM T64567 C5HM8E 474578 Ki = 78.7 nM T64567 CL0M9Y 482317 Ki = 10500 nM T64567 CHF2Y9 493949 Ki = 403 nM T64567 C02DMG 504302 Ki = 10.1 nM T64567 CU7XE2 504303 Ki = 51.4 nM T64567 CNLT49 504304 Ki = 35 nM T64567 COGF52 516871 Ki = 130000 nM T64567 C49CNT 519869 Ki = 810 nM T64567 CU8MR5 520660 Ki = 1350 nM T64567 C5OA7L 522689 Ki = 48000000 nM T64567 CJ7FR6 533728 Ki = 1413 nM T64567 C24ASH 539731 Ki = 53.8 nM T64567 C7EBA4 540544 Ki = 44.9 nM T64567 CFU6X9 560256 Ki = 714 nM T64567 CPV28T 567846 Ki = 184 nM T64567 CGHE12 607195 Ki = 330 nM T64567 CIK9S3 607305 Ki = 209 nM T64567 CP3SF2 609637 Ki = 54500 nM T64567 C5EA3O 638001 Ki = 7450 nM T64567 C1DX6J 640625 Ki = 19600 nM T64567 CUMO27 643477 Ki = 3380 nM T64567 C58QOW 643497 Ki = 31 nM T64567 CH05FZ 648662 Ki = 26.6 nM T64567 C6PTC3 658040 Ki > 50000 nM T64567 CS9F8K 667829 Ki = 1120 nM T64567 CRTE89 667830 Ki = 317 nM T64567 CU9ZY6 670087 Ki = 72.5 nM T64567 CYGK68 676946 Ki = 610 nM T64567 CF9V6Q 699414 IC50 = 850000 nM T64567 C4YWI2 702292 Ki = 4.5 nM T64567 CYZ9O5 703304 Ki = 51.4 nM T64567 C9JH0M 706033 Ki = 150 nM T64567 C7ZE6K 706849 Ki > 50000 nM T64567 CK7DO5 708535 Ki = 37 nM T64567 CK9HY0 716763 Ki = 5.9 nM T64567 C8J4SO 724642 Ki = 40 nM T64567 C61NGE 724799 Ki = 2.4 nM T64567 C8J7CO 730546 Ki = 32.1 nM T64567 C8G7EC 730672 Ki = 58 nM T64567 CNJZ35 738819 Ki > 50000 nM T64567 CV6Y7U 740560 IC50 = 79 nM T64567 CZM6W0 742873 Ki = 4.4 nM T64567 CLG6H5 746816 Ki = 39.9 nM T64567 CRIJ01 747569 Ki = 21 nM T64567 CW90GV 767467 Ki = 41.6 nM T64567 CV79DU 776418 Ki > 50000 nM T64567 CQJ06V 780268 IC50 = 2.86 nM T64567 CO1KN3 788171 Ki = 4.3 nM T64567 CA2B8X 792066 Ki = 47.9 nM T64567 CM0VX3 809685 Ki = 12.6 nM T64567 C6LN8S 816982 Ki = 5470 nM T64567 C5BGW9 818267 Ki > 50000 nM T64567 CJP5D4 818647 IC50 = 90 nM T64567 CVJZ57 818753 Ki = 310 nM T64567 CF93TC 821388 Ki = 820 nM T64567 C5VJZ0 822776 Ki = 0.32 nM T64567 CTD64N 834412 Ki = 2.2 nM T64567 CHE97G 834460 IC50 = 341.71 nM T64567 C51FVL 906840 Ki = 17.5 nM T64567 CKV7B6 917551 Ki = 19 nM T64567 C4I3PJ 922062 Ki = 5.3 nM T64567 CRGQ70 927433 Ki = 390 nM T64567 CO7XW0 928228 Ki = 40.2 nM T64567 C6XQO2 940540 Ki > 50000 nM T64567 C4L9QD 943114 Ki = 30 nM T64567 COH62A 943115 Ki = 29.3 nM T64567 CX3U0S 975396 Ki > 50000 nM T64567 CZ3WK7 983751 Ki = 4.4 nM T64567 CN71CV 989611 Ki = 22 nM T64567 C5CED0 1014382 IC50 = 0.12 nM T64567 CXQ3M7 1016209 IC50 = 3.11 nM T64567 C6MU1W 1069008 Ki = 300 nM T64567 CJ2S0M 1070919 Ki = 9.5 nM T64567 CYS9A2 1070922 Ki = 32.6 nM T64567 CM2C5N 1070928 Ki = 21.2 nM T64567 COM2R4 1070933 Ki = 35.6 nM T64567 CKA4R5 1080680 Ki = 1070 nM T64567 CDK1Z2 1085887 Ki = 49500 nM T64567 CA67JK 1124687 Ki = 4.9 nM T64567 CZ04BL 1136487 IC50 = 21.64 nM T64567 CWD7G1 1147802 Ki = 290 nM T64567 CJ82NF 1178394 Ki = 9.6 nM T64567 C7A8VI 1211699 Ki = 350 nM T64567 CYF34N 1211700 Ki = 428 nM T64567 C7QP5E 1213792 Ki = 8.1 nM T64567 CL87AM 1286568 Ki = 257 nM T64567 CA1I9S 1286583 Ki = 360 nM T64567 CE6W7O 1287222 Ki = 23.6 nM T64567 CP60YD 1294363 Ki = 9.3 nM T64567 CYGO97 1300832 IC50 = 3.42 nM T64567 C5XNB4 1307068 Ki = 84.7 nM T64567 CDWO53 1346695 Ki = 1.2 nM T64567 CC3G1N 1377410 Ki = 36 nM T64567 CN5I0K 1505151 Ki = 200 nM T64567 CAHP42 1548275 Ki = 171 nM T64567 C51SMF 1551768 Ki = 970 nM T64567 CORY25 1581900 Ki = 23.78 nM T64567 C4YUX5 1594254 Ki = 2750 nM T64567 C40YCV 1655994 Ki = 126.2 nM T64567 CU7KR6 1738244 Ki = 102 nM T64567 C7XSO5 1748172 Ki = 89.7 nM T64567 CGKP07 1748225 Ki = 17.7 nM T64567 C98OLG 1775694 Ki = 23 nM T64567 C5PU0O 1809247 IC50 = 14.95 nM T64567 C9ZEH2 1825978 IC50 = 10.42 nM T64567 CTF8R5 1957305 Ki = 2510 nM T64567 CR56WH 1968441 IC50 = 0.47 nM T64567 C1DWG0 1989902 Ki = 9.2 nM T64567 CDQR23 2049187 Ki = 10.1 nM T64567 CSQJ97 2065546 Ki = 2078 nM T64567 CTK8C6 2089520 Ki = 240 nM T64567 C93VNU 2089779 Ki = 1169 nM T64567 C3W4PG 2192287 Ki = 3 nM T64567 CQS3A7 2207483 Ki = 122.8 nM T64567 C3Z4RX 2278691 IC50 = 17950 nM T64567 CEW2Q3 2283723 Ki = 3370 nM T64567 COB96D 2305168 Ki = 1220 nM T64567 C6FN0O 2316976 Ki = 296 nM T64567 CGW6L4 2318645 Ki = 4470 nM T64567 CD98QK 2333105 Ki = 980 nM T64567 C1V0KL 2357187 Ki = 5.2 nM T64567 C3BJ4K 2368995 Ki = 138 nM T64567 CTJ42W 2368997 Ki = 39.1 nM T64567 C4TD8M 2388085 Ki = 3.3 nM T64567 C1TW9F 2457081 Ki = 539 nM T64567 CR65UH 2471990 Ki > 50000 nM T64567 C95INQ 2476733 Ki = 0.3 nM T64567 C75SLD 2496330 Ki = 0.25 nM T64567 C2H4KT 2520594 Ki = 8.9 nM T64567 CKH53Q 2723810 Ki = 1220000 nM T64567 C8YH7W 2733779 Ki = 370 nM T64567 C0V7XB 2733782 Ki = 9.2 nM T64567 C0W8UL 2735045 Ki = 566 nM T64567 CQ70UR 2755708 Ki = 2.1 nM T64567 CU60ZB 2755709 Ki = 2.2 nM T64567 CNG69U 2755712 Ki = 2.4 nM T64567 C58ISM 2755728 Ki = 2.9 nM T64567 CD41AE 2795990 Ki = 196 nM T64567 CCOI52 2797418 Ki = 22 nM T64567 CPO6W3 2813478 Ki = 6.2 nM T64567 CUI4Y8 2814914 Ki = 23 nM T64567 CLFB40 2815883 Ki = 139.1 nM T64567 CDSN81 2826269 Ki = 0.32 nM T64567 CEY4J6 2858793 IC50 = 198.98 nM T64567 CU6D3W 2881615 IC50 > 3900 nM T64567 CBPO81 2882281 Ki = 26 nM T64567 CVA6F2 2893744 IC50 = 0.48 nM T64567 CE2GR3 2900806 Ki = 12200 nM T64567 CW9M7A 2952488 Ki = 91 nM T64567 CFO90D 2952737 Ki = 380 nM T64567 CFV92S 3000601 Ki = 973 nM T64567 CZEH20 3003616 Ki = 40.8 nM T64567 CJ9LZ7 3051101 Ki = 1350 nM T64567 CN2Y5M 3083616 Ki = 850 nM T64567 C9GT5Z 3083928 Ki = 6580 nM T64567 C84TYH 3108089 IC50 = 28.35 nM T64567 CY19CS 3115791 Ki = 884 nM T64567 C49VDN 3132886 Ki = 760 nM T64567 CQI7A2 3133127 Ki = 8654 nM T64567 CXU4J8 3377675 Ki = 4.7 nM T64567 C1K6IA 3379075 Ki = 3.1 nM T64567 CL6E2Y 3426384 Ki = 933.6 nM T64567 CIS69V 3440976 Ki = 56.5 nM T64567 CT1NB8 3441996 Ki = 7.8 nM T64567 CZW71J 3476048 IC50 = 0.48 nM T64567 CIXH89 3516083 Ki = 8.5 nM T64567 C0VI6O 3524248 Ki = 42000 nM T64567 CKTY04 3538605 Ki = 70.4 nM T64567 C86GSL 3542746 Ki = 8.7 nM T64567 CHGS79 3551941 Ki = 24.8 nM T64567 C9L1HS 3586494 Ki = 3.8 nM T64567 C4WZG2 3657160 Ki = 11 nM T64567 C3REH6 3703019 IC50 = 70 nM T64567 CQ5F9P 3724005 Ki = 8.1 nM T64567 C1JU9P 3774719 Ki = 51.3 nM T64567 C2SY4L 3856570 Ki = 37.6 nM T64567 CI3KT8 3936209 Ki = 61.3 nM T64567 CJ6D2S 3970972 Ki = 0.53 nM T64567 C8DZ4B 4121769 Ki = 8.2 nM T64567 CT57HM 4204917 Ki = 23 nM T64567 CV6BJ7 4262171 Ki = 55.1 nM T64567 CUT26E 4274816 Ki = 45000 nM T64567 CUE97L 4276695 Ki = 20.6 nM T64567 CI6AE7 4377996 Ki = 271000 nM T64567 CJ63TI 4578038 Ki = 0.45 nM T64567 CE5LO8 4578265 Ki = 173.6 nM T64567 C7RS2F 4583704 Ki = 22.1 nM T64567 CAPM27 4598704 Ki = 48000 nM T64567 CLSY09 4626049 Ki = 780 nM T64567 CLQ7U4 4627354 IC50 = 4.14 nM T64567 CPX3W6 4650747 Ki = 243 nM T64567 CTM71V 4654716 Ki = 198 nM T64567 C07MRI 4712722 Ki = 100000 nM T64567 CWXE71 4718084 Ki = 4.3 nM T64567 C6RC3L 4718087 Ki = 10.2 nM T64567 C5FZ0L 4718107 IC50 = 18.81 nM T64567 CRL7B4 4718142 Ki = 2.9 nM T64567 CJM5F3 4718971 Ki = 4.3 nM T64567 CAG10X 4723337 IC50 = 68.46 nM T64567 C6B0OY 4723880 Ki = 3.5 nM T64567 C0MFT8 4801151 Ki = 221 nM T64567 CSC7B8 4803242 Ki = 3.7 nM T64567 CUA65R 4857564 Ki = 62.5 nM T64567 CX8C3P 4961927 Ki = 235 nM T64567 CX3RJ9 5005133 Ki = 72.1 nM T64567 CRQ2H5 5010026 IC50 = 26150 nM T64567 CIP6Q8 5017140 Ki = 0.21 nM T64567 CF94ER 5032527 Ki = 19 nM T64567 C49FDN 5046067 Ki = 107.9 nM T64567 C4OAL9 5070078 Ki = 4700 nM T64567 CN31CX 5071527 Ki = 8.4 nM T64567 CU8E4B 5133468 Ki = 210 nM T64567 C7GXU1 5147921 Ki = 8100000 nM T64567 CM9N8G 5161767 Ki = 94.7 nM T64567 C6HM0R 5164092 Ki = 9510 nM T64567 C4HB1G 5172319 Ki = 8.3 nM T64567 CI8JY0 5172475 Ki = 30 nM T64567 CFQ62G 5232078 Ki > 100000 nM T64567 CEBD92 5272990 Ki = 8400 nM T64567 CP09FG 5272997 Ki > 100000 nM T64567 C4SV5T 5273568 Ki = 370 nM T64567 CU4E5S 5273569 Ki = 610 nM T64567 CZS0G5 5276565 IC50 > 10000 nM T64567 C3JN0F 5277465 IC50 > 10000 nM T64567 CRJK67 5277481 IC50 > 10000 nM T64567 CYF7S5 5277490 IC50 > 10000 nM T64567 CD1LZ7 5278580 Ki = 0.9 nM T64567 CNZ73E 5280567 Ki = 560 nM T64567 CA18OQ 5316302 Ki = 850 nM T64567 CTJ01E 5317485 Ki = 3500 nM T64567 CI58XK 5319562 Ki = 850 nM T64567 CNO53D 5321265 Ki = 620 nM T64567 CP0R5H 5336569 Ki = 39.5 nM T64567 C8PS4E 5358858 Ki = 4030 nM T64567 C4KHR2 5431473 IC50 = 19.09 nM T64567 CH5OM1 5463917 Ki = 42600000 nM T64567 CXEW32 5491996 Ki = 3220 nM T64567 C7RG3L 5496307 Ki = 6790 nM T64567 CX71JE 5682293 Ki = 20.3 nM T64567 CWYU91 5742696 Ki = 6930 nM T64567 CU0FW5 5743063 Ki = 8280 nM T64567 C4VZP8 5765787 Ki = 0.93 nM T64567 CWL5R2 5765789 Ki = 5.4 nM T64567 CK0M4A 5910585 Ki = 600 nM T64567 CHJ3V8 6102658 Ki = 220 nM T64567 CMD1Q0 6460079 Ki = 6.7 nM T64567 CS4KQ6 6482974 Ki = 760 nM T64567 C9L8AX 6537802 Ki = 58 nM T64567 C65FRB 6852128 Ki = 1.3 nM T64567 CK85ZF 7022526 IC50 = 74 nM T64567 C0W5GD 7130726 Ki = 8.7 nM T64567 CWL9C2 7382212 Ki = 234 nM T64567 C75SBG 7382231 Ki = 390 nM T64567 C6U9MT 7382238 Ki > 50000 nM T64567 CY57CX 7382249 Ki = 616 nM T64567 CKCM96 7463376 Ki = 3400 nM T64567 CDCP43 7766335 Ki = 1030 nM T64567 CTH8D3 7785988 Ki = 1245 nM T64567 C95AKP 7794397 Ki = 184 nM T64567 C6S5HK 7832430 Ki = 878 nM T64567 C1EKW8 7996519 Ki = 55.9 nM T64567 C67SFK 8084575 Ki = 360 nM T64567 CQ0Z4E 8098235 Ki = 34 nM T64567 CSW01Z 8272034 Ki = 191 nM T64567 C9BAM4 8281641 Ki = 20.5 nM T64567 C3WQ9M 8866559 Ki = 0.96 nM T64567 C5CS1Y 9314410 Ki = 11.6 nM T64567 C3SA2N 9314413 Ki = 2 nM T64567 C47VSJ 9572721 Ki > 10000 nM T64567 CIJ25V 9794947 IC50 = 6080 nM T64567 C7SRM4 9837496 IC50 = 8890 nM T64567 C0EJ1Q 9847197 Ki = 16 nM T64567 CSIY73 9952009 IC50 > 100000 nM T64567 CJS4I3 9990000 Ki = 14 nM T64567 CIN68V 9998184 Ki = 0.34 nM T64567 CY47OI 9998322 Ki = 24 nM T64567 CXD28H 10015065 Ki = 19 nM T64567 CNKD31 10016330 Ki = 73.3 nM T64567 C4UEV9 10016475 Ki = 33.3 nM T64567 CF6RN0 10018880 Ki = 0.15 nM T64567 CX2W9O 10037048 IC50 = 8120 nM T64567 C5X7GY 10059582 Ki = 367.6 nM T64567 C69DPZ 10068042 IC50 = 397 nM T64567 CY8F0E 10076040 Ki = 6330 nM T64567 C0P5XV 10081897 Ki = 45.8 nM T64567 CD58EL 10083644 Ki = 860 nM T64567 CRN29P 10104483 Ki = 18 nM T64567 C7WU0A 10107532 Ki = 31 nM T64567 CAQ6I1 10131078 Ki = 15 nM T64567 CXD91O 10136406 Ki = 12.9 nM T64567 CVRZ27 10198038 IC50 = 8970 nM T64567 C63AZQ 10198750 Ki = 13 nM T64567 CUR4O7 10198795 Ki = 10 nM T64567 CJV68L 10220266 Ki = 28.2 nM T64567 C4E1JQ 10245883 Ki = 20 nM T64567 CLM6Z5 10290835 Ki > 1000 nM T64567 CN40WD 10331524 Ki = 56.9 nM T64567 CUE81P 10337354 Ki = 51 nM T64567 C3HBY6 10375558 Ki = 22 nM T64567 CT9VJ3 10383097 Ki = 15.2 nM T64567 C1O2FH 10383098 Ki = 0.8 nM T64567 CP2XW6 10387325 Ki = 8 nM T64567 CVW18K 10409391 Ki = 71 nM T64567 C5IK7H 10420920 Ki = 36 nM T64567 C4MI8O 10423003 Ki = 9 nM T64567 CFGK83 10430595 Ki = 4.3 nM T64567 C6TYP0 10467861 Ki = 116.2 nM T64567 C25NJB 10471772 Ki = 27 nM T64567 C13JVK 10477954 Ki = 31 nM T64567 CU8E4S 10505384 Ki = 160 nM T64567 CRS2V1 10505991 Ki = 450 nM T64567 CH6A2O 10507009 Ki = 84 nM T64567 CD41CA 10512636 Ki = 415.9 nM T64567 CU6HX8 10530223 Ki = 37 nM T64567 C6C7YQ 10531119 Ki = 120 nM T64567 CA5C0S 10531121 Ki > 500 nM T64567 C8CJ3W 10554523 Ki = 70 nM T64567 CT6BA5 10572515 Ki = 72 nM T64567 CF3A4I 10577600 Ki = 100 nM T64567 C73KXU 10586607 Ki = 6200 nM T64567 CAZ36G 10596413 Ki = 29 nM T64567 CO8D2C 10602116 Ki = 89 nM T64567 C97JCY 10625036 Ki = 178 nM T64567 CU3YT8 10625038 Ki = 8 nM T64567 C4FLA9 10625484 Ki = 230 nM T64567 CGI03J 10625651 Ki = 81 nM T64567 CGB5S0 10626619 Ki = 78 nM T64567 C9TSQ6 10632698 Ki = 5100 nM T64567 CQB3T1 10650115 Ki = 3 nM T64567 CC4UM6 10650450 Ki > 500 nM T64567 C1W7CO 10671070 Ki = 54 nM T64567 CETF96 10673746 Ki > 500 nM T64567 CVHO36 10692638 Ki = 146 nM T64567 C2YH7O 10696741 Ki = 280 nM T64567 CRL2U7 10696743 Ki = 106 nM T64567 CE82AF 10697359 Ki = 205 nM T64567 C1P2SH 10698664 Ki = 95 nM T64567 C6D2TJ 10712038 Ki = 4580 nM T64567 CX8YI4 10716240 Ki = 35 nM T64567 CNF6H0 10721639 Ki > 500 nM T64567 C2ZLE4 10737428 Ki = 5.1 nM T64567 C7WHI1 10745371 Ki = 135 nM T64567 CB7T3Q 10755646 Ki = 964 nM T64567 C3HVQ9 10764510 Ki = 42 nM T64567 CH78WD 10766083 Ki = 26 nM T64567 CIB3E5 10766650 Ki = 43 nM T64567 C06MYS 10766652 Ki = 6 nM T64567 C7X3PW 10768529 Ki > 500 nM T64567 CHVB87 10768870 Ki = 80 nM T64567 CDO17N 10792606 Ki > 500 nM T64567 C5Q0HP 10792608 Ki = 85 nM T64567 CQR74O 10813858 Ki = 49 nM T64567 C9S1KI 10816020 Ki = 79 nM T64567 CLS5J3 10836786 Ki = 48 nM T64567 C32QME 10838459 Ki = 29 nM T64567 C7DV4E 10868086 Ki = 33 nM T64567 CQN7G6 10869299 Ki = 69 nM T64567 CT0KQ8 10878827 Ki = 12 nM T64567 C3WOS1 10917392 Ki = 11500 nM T64567 C6EPH9 10919571 Ki = 9.6 nM T64567 C8CV1Z 10923837 Ki = 37 nM T64567 CL5D1P 10926842 Ki = 310000 nM T64567 C3WN6P 10931938 Ki = 531 nM T64567 C7FP4E 10932133 Ki = 6.2 nM T64567 CGI4X1 10933094 Ki = 23.4 nM T64567 CD3GB7 10937101 Ki = 46 nM T64567 CN27BY 10953838 Ki = 970 nM T64567 CIXO05 10959593 Ki = 46 nM T64567 CEV7Z1 10962037 Ki = 39 nM T64567 CQO1E7 10962986 Ki = 41 nM T64567 C73HZT 10983658 Ki = 21 nM T64567 CCIT95 11003980 Ki = 24 nM T64567 C1D7XA 11011569 Ki = 33 nM T64567 C9IF1C 11013393 Ki = 39 nM T64567 CD4JQ1 11015176 Ki = 47 nM T64567 CAED68 11021701 Ki = 47 nM T64567 CDB16V 11026415 Ki = 27 nM T64567 CD8HS3 11031678 Ki = 45 nM T64567 CWO84N 11032771 Ki = 51 nM T64567 C36BAC 11034581 Ki > 100000 nM T64567 CN6QX1 11036198 Ki = 86 nM T64567 CV75NH 11047521 Ki = 79 nM T64567 CQBP46 11061197 Ki = 7.3 nM T64567 C8C6ER 11069133 Ki = 38 nM T64567 COGV98 11074431 Ki = 2400 nM T64567 CMK4Y0 11096006 Ki = 19.1 nM T64567 CWB10K 11103986 Ki = 7.9 nM T64567 CVZ89X 11112315 Ki = 96800 nM T64567 CYQ01S 11115351 Ki = 7.5 nM T64567 CH6IE3 11117198 Ki = 28.2 nM T64567 C8X2DC 11127784 Ki = 53 nM T64567 C6RM4H 11134231 Ki = 78 nM T64567 C5WS3E 11147931 IC50 = 8300 nM T64567 CP3CU4 11157709 Ki = 6 nM T64567 CC4IE1 11158128 Ki = 24 nM T64567 CPB0A5 11164855 Ki = 3.2 nM T64567 C50HJY 11177131 Ki = 7.9 nM T64567 CIL4M9 11183499 Ki > 100000 nM T64567 C4W0YX 11186322 Ki = 22 nM T64567 C31DIQ 11188711 Ki = 76 nM T64567 C2CHY5 11188898 Ki = 750 nM T64567 C5C6MG 11194613 Ki > 1000 nM T64567 C5Y1CV 11196316 Ki > 1000 nM T64567 C75FMT 11199252 Ki = 9.5 nM T64567 CFG37K 11209006 Ki = 22 nM T64567 C0P8JA 11215523 Ki = 32 nM T64567 C2AFO0 11216333 Ki = 20 nM T64567 C5L7NR 11217340 Ki = 633 nM T64567 CY2VA5 11221764 Ki = 9.5 nM T64567 CY1P4Q 11223689 Ki = 8.6 nM T64567 CY9W5K 11226359 Ki = 7.6 nM T64567 C39QJA 11234047 Ki = 10.5 nM T64567 CXAS45 11235150 Ki = 8.5 nM T64567 C8O1FM 11239393 Ki = 32 nM T64567 CHC42Y 11245700 Ki = 18 nM T64567 CGE40M 11245996 Ki = 5.4 nM T64567 CCLV87 11247335 Ki = 7.9 nM T64567 CN86YV 11250791 Ki = 16 nM T64567 CI7YT0 11252120 Ki > 1000 nM T64567 C7UVW8 11258440 Ki = 5.8 nM T64567 C12URI 11261582 Ki = 5 nM T64567 CIR6A0 11262484 Ki = 40 nM T64567 C7FA3C 11274029 Ki = 43 nM T64567 CCSA87 11280465 Ki = 162 nM T64567 CF15AS 11287957 Ki = 98.7 nM T64567 C0H6GB 11292444 Ki = 8.5 nM T64567 C1FJ7I 11304583 Ki = 64 nM T64567 C3CDO1 11309586 Ki = 631 nM T64567 CRP08M 11310883 IC50 = 6360 nM T64567 CBC47W 11312414 Ki = 15 nM T64567 CAU4B5 11317320 Ki = 24 nM T64567 CB4U3M 11318985 Ki = 29 nM T64567 CHA0V5 11321514 Ki = 800 nM T64567 C8ZA1X 11326347 Ki = 7.3 nM T64567 CU73JN 11339017 Ki = 6.2 nM T64567 C8Q5VJ 11342941 Ki = 40 nM T64567 CV80KU 11346010 Ki = 16700 nM T64567 CCY4G5 11350445 Ki = 83 nM T64567 C3NGH2 11352609 Ki = 3.2 nM T64567 C8PM3Z 11353795 Ki = 24 nM T64567 C8MI3Z 11361075 Ki = 16 nM T64567 CY3B6F 11362509 Ki = 72 nM T64567 CM8Y1J 11367571 IC50 = 8260 nM T64567 CM1XU5 11373291 Ki = 32 nM T64567 C6QO0H 11384370 Ki = 7 nM T64567 CY64KU 11385765 Ki = 13 nM T64567 CIQ5K7 11387799 Ki = 16 nM T64567 C7MK2E 11390955 Ki = 279 nM T64567 CVT2K6 11396353 Ki = 5.4 nM T64567 CT3E0Y 11399060 Ki = 30 nM T64567 C6RUJ7 11399350 Ki = 15 nM T64567 CEO47P 11399506 Ki = 35 nM T64567 CH98MP 11399715 Ki = 29 nM T64567 CBVL07 11407223 Ki = 5.4 nM T64567 C3KV6R 11407281 Ki = 70 nM T64567 C8DF5O 11416806 Ki = 120 nM T64567 CG1A5D 11427826 Ki = 1840 nM T64567 CGPE75 11428235 Ki = 12.6 nM T64567 CT3NI0 11433608 Ki = 9 nM T64567 C3KRG4 11433767 Ki = 35 nM T64567 CUR65I 11441308 Ki = 15 nM T64567 CTU87D 11441601 Ki = 13 nM T64567 C7EOG0 11441729 Ki = 4.8 nM T64567 C41CHM 11445520 Ki = 16 nM T64567 CMS0Q5 11445529 Ki = 12 nM T64567 C4BQM5 11455128 Ki = 5.5 nM T64567 C2J9BG 11463026 Ki = 8.3 nM T64567 CFER43 11467281 Ki = 26 nM T64567 CM9I6W 11467962 Ki = 30 nM T64567 CQ1D6E 11470070 IC50 = 8590 nM T64567 C91XWJ 11478542 Ki = 34 nM T64567 CIWG06 11479385 Ki = 12 nM T64567 CCY54I 11479559 Ki = 45 nM T64567 CL1RC2 11485376 Ki = 24 nM T64567 CQ9H8J 11490915 Ki = 31 nM T64567 CNFY48 11514219 Ki = 306000 nM T64567 CU8YH7 11533895 Ki = 24 nM T64567 CP8AX2 11540662 Ki = 5 nM T64567 CIMD40 11578176 Ki = 6860 nM T64567 CUJI91 11581618 Ki = 165 nM T64567 CDS25O 11593765 IC50 = 8600 nM T64567 CCB82K 11596108 Ki = 1725 nM T64567 C9QL2F 11615432 Ki = 139.5 nM T64567 C36MZP 11616716 Ki = 3.1 nM T64567 C4EC3U 11663528 Ki = 64 nM T64567 C95PYS 11667431 Ki = 16 nM T64567 C9JR2I 11674590 Ki = 17400 nM T64567 CRG49U 11674754 Ki = 2.8 nM T64567 CPGO32 11675510 Ki = 38 nM T64567 C7ZPR9 11681852 Ki = 1.3 nM T64567 CCG17H 11688636 Ki = 1.5 nM T64567 CF8IT6 11696964 Ki = 21 nM T64567 C4VZO5 11709992 Ki = 208 nM T64567 CHAN30 11714982 Ki = 21 nM T64567 C5QIK4 11721174 Ki = 120 nM T64567 CAW47S 11733056 Ki = 23 nM T64567 CP78CU 11763512 Ki = 34 nM T64567 CWM5I6 11773896 Ki = 35 nM T64567 CV68TJ 11774586 Ki = 7 nM T64567 CH7Q5S 11777250 Ki = 7.9 nM T64567 C37CKB 11782720 Ki = 43 nM T64567 C6S8WR 11786209 Ki = 5 nM T64567 C4BH9A 11788388 Ki = 386 nM T64567 CV7HN1 11795548 Ki = 14 nM T64567 CSD5K9 11806775 Ki = 54 nM T64567 C0RZ9Y 11816502 Ki = 12 nM T64567 C8DY3Z 11817193 IC50 = 9140 nM T64567 C73SVE 11817275 Ki = 7.8 nM T64567 CTR0U7 11823783 Ki = 63 nM T64567 C45NRP 11851425 Ki = 471 nM T64567 CQXG94 11970596 Ki = 3060000 nM T64567 CZD0B3 11974341 Ki = 430 nM T64567 C27HSO 11974343 Ki = 135 nM T64567 CCM17V 11974451 Ki = 360 nM T64567 CX4IJ0 11974452 Ki = 238 nM T64567 C59UEI 11974453 Ki = 1100 nM T64567 CYS7X0 11974454 Ki = 204 nM T64567 C09JGZ 11974455 Ki = 132 nM T64567 CS9VL2 11974456 Ki = 1200 nM T64567 CP39YI 11974558 Ki = 125 nM T64567 CB97SM 11974559 Ki = 54 nM T64567 CE8WN6 11974560 Ki = 65 nM T64567 C06CBY 11974561 Ki = 108 nM T64567 CU6K0N 11974562 Ki = 39 nM T64567 CI7OE1 11974563 Ki = 76 nM T64567 C6Z5DX 11974630 Ki = 124 nM T64567 CW4X9G 11974631 Ki = 221 nM T64567 CEBO65 11974632 Ki = 1238 nM T64567 CGQ6B7 11974724 Ki = 130 nM T64567 CHO9T1 11974725 Ki = 442 nM T64567 CC8TS1 11974727 Ki = 23 nM T64567 CDL18J 11974728 Ki = 183 nM T64567 C7G3YS 11974830 Ki = 241 nM T64567 C1C4JW 11974831 Ki = 67 nM T64567 CXW89D 12004261 Ki = 32 nM T64567 C0L4OC 12049163 Ki = 4370 nM T64567 C4ZYQ1 12049713 Ki = 890000 nM T64567 CMPA32 12066940 Ki > 500000 nM T64567 CB15KR 12066941 Ki > 500000 nM T64567 C2XBZ3 12070806 Ki = 92 nM T64567 C32TWU 12094253 Ki = 44.5 nM T64567 C6P1VC 12188108 Ki > 10000 nM T64567 C3C9ON 12226066 Ki = 930 nM T64567 CCY51E 12237458 Ki = 123.1 nM T64567 C18LXJ 12411101 Ki = 59 nM T64567 C0C8FG 12411107 Ki = 50 nM T64567 CLB1E3 12499681 Ki = 28.4 nM T64567 CP87GR 12516475 Ki = 12.8 nM T64567 C5RS4H 12528487 Ki = 63.9 nM T64567 CM8TP6 12528490 Ki = 35.8 nM T64567 C35CMO 12589789 Ki = 35.8 nM T64567 CZCF65 12914626 Ki > 1000 nM T64567 C1GNM5 12914627 Ki > 1000 nM T64567 CO8WC5 12938307 Ki = 8.5 nM T64567 CP70LE 12954894 Ki = 246 nM T64567 C4IKA3 13087489 Ki = 1005 nM T64567 CF2BM7 13177311 Ki = 2.6 nM T64567 C8VM1A 13201770 Ki = 680 nM T64567 CV1UF4 13306723 Ki = 57.1 nM T64567 C85GSD 13360355 Ki = 458 nM T64567 C79BND 13361840 Ki = 90590 nM T64567 CX7M9C 13373975 Ki = 40.3 nM T64567 CHC41Q 13381193 Ki = 59 nM T64567 COLK69 13419352 Ki = 26.3 nM T64567 C3HOK8 13580495 Ki > 1000 nM T64567 CFN29Y 13584466 Ki = 41.4 nM T64567 CQTX49 13738810 IC50 > 10000 nM T64567 CTYP72 13949092 Ki = 22.2 nM T64567 CR6HB5 13949095 Ki = 402.8 nM T64567 CFMK94 13949102 Ki = 40.2 nM T64567 C7K4JV 14024589 Ki = 273.4 nM T64567 C4UG2O 14057643 Ki = 670 nM T64567 CLS53V 14151811 IC50 = 95 nM T64567 CQ3D9C 14151815 IC50 = 200 nM T64567 CNZ6H2 14205726 Ki = 7900000 nM T64567 C92OEB 14498136 Ki = 13.9 nM T64567 CHOG93 14611919 Ki = 102 nM T64567 CZ6SN8 14777102 Ki = 77.9 nM T64567 C35DGV 14873166 Ki = 8.5 nM T64567 C9CLH4 14873170 Ki = 27.1 nM T64567 C9K0LX 14873174 Ki = 25.2 nM T64567 CM34ER 14873177 Ki = 35.8 nM T64567 C7XD2T 15118768 Ki = 780 nM T64567 CK8GE9 15230629 Ki = 408.5 nM T64567 C6F3GK 15267134 Ki = 23.64 nM T64567 CDE4F9 15290967 Ki = 38.4 nM T64567 CW72MS 15438999 Ki = 97 nM T64567 C7R5AH 15476112 Ki = 210 nM T64567 C3CTS0 15523879 Ki = 1 nM T64567 C2G4FH 15599374 Ki = 6.1 nM T64567 CT73PL 15618966 Ki = 2.1 nM T64567 CLIO60 15645619 Ki = 216.1 nM T64567 CLT47Z 15783680 Ki = 4747.6 nM T64567 C6F0XZ 15818962 Ki = 563 nM T64567 C8PER5 15938557 Ki > 500000 nM T64567 CB3S7I 16007202 Ki = 6.9 nM T64567 CM06OZ 16046226 Ki = 14.5 nM T64567 CVZG29 16072592 Ki = 16230 nM T64567 CB73ST 16072595 Ki = 15100 nM T64567 C6U0VS 16078349 Ki = 48 nM T64567 CUT32D 16078350 Ki > 1000 nM T64567 C4JIO0 16078351 Ki = 37 nM T64567 C23FGI 16078837 Ki = 4190 nM T64567 CQ0UX9 16082752 Ki = 78 nM T64567 CBRL45 16082753 Ki = 72 nM T64567 C0BIQ3 16082754 Ki = 18 nM T64567 C6KN4Z 16082755 Ki = 9.3 nM T64567 C94FZV 16082756 Ki = 79 nM T64567 C85HIK 16082757 Ki = 71 nM T64567 CC74NH 16087011 Ki = 8.3 nM T64567 C1CD5B 16087012 Ki = 8.1 nM T64567 C8AP5W 16087015 Ki = 7.9 nM T64567 CLNI97 16087025 Ki = 8.3 nM T64567 CBWD20 16087028 Ki = 7 nM T64567 CN1XR0 16087029 Ki = 58.8 nM T64567 C3GMJ8 16087031 Ki = 6.9 nM T64567 CC0Z4V 16119626 Ki = 710 nM T64567 CV5O8W 16125524 Ki = 101 nM T64567 CZ7T4C 16125526 Ki = 107 nM T64567 CS78TE 16125527 Ki = 9.7 nM T64567 C1Z9GQ 16125580 Ki = 345 nM T64567 CE4SB2 16125581 Ki = 120 nM T64567 CWM0L9 16125582 Ki = 69 nM T64567 C4SD3N 16125583 Ki = 84 nM T64567 CN03IT 16227153 Ki = 50.5 nM T64567 CGB45O 16235229 Ki = 409 nM T64567 CG7OL3 16693908 Ki = 18500000 nM T64567 CMB87O 16717602 Ki = 4.5 nM T64567 COQU32 16729004 Ki = 8.1 nM T64567 CTK68M 17249579 Ki = 7 nM T64567 C5DT7E 17250082 Ki = 5.1 nM T64567 C6THW2 17268490 Ki = 541 nM T64567 C5CE8Z 17371280 Ki = 0.86 nM T64567 CA4OE9 17371576 Ki = 0.67 nM T64567 C73YML 17385730 Ki = 199 nM T64567 C91LAN 17413757 Ki = 165 nM T64567 C5M9DR 17433209 Ki = 50.9 nM T64567 CYLM41 17492191 Ki > 10000 nM T64567 CDWU20 17537594 Ki = 53.2 nM T64567 CUP95O 17562622 Ki = 4.8 nM T64567 CK7D2I 17748220 Ki = 110 nM T64567 C3AX8E 17774014 Ki = 296 nM T64567 C6SFI8 18268734 Ki = 122.2 nM T64567 CR9VF3 18668331 Ki = 13.5 nM T64567 C60NAV 18971452 Ki = 12.6 nM T64567 C2K5BX 19374444 Ki = 17.9 nM T64567 CIEH93 19382975 IC50 > 10000 nM T64567 C62PKT 19838794 Ki = 28.2 nM T64567 CU3QS7 19898674 Ki = 58.8 nM T64567 CB46JX 20109894 Ki = 7790 nM T64567 CGE35Q 20182298 Ki = 3.7 nM T64567 CXJ2H4 20195196 Ki = 6830 nM T64567 C8Z1CM 20216502 Ki = 126 nM T64567 CAG0O1 20368972 Ki = 2020 nM T64567 C15BEG 20694083 Ki = 41.4 nM T64567 CF28QV 21017876 Ki = 1150 nM T64567 CCJ8Q3 21051266 Ki = 25.6 nM T64567 CH15RE 21051367 Ki = 69.1 nM T64567 CV34MD 21149346 Ki = 40 nM T64567 CJGU80 21240387 Ki = 23.9 nM T64567 C18KAH 21297028 Ki = 76.1 nM T64567 C9J1WT 21497848 Ki = 481 nM T64567 CC5W7X 21542156 Ki = 436 nM T64567 CD0K1C 21600238 Ki = 23.1 nM T64567 C61KUX 21726402 Ki = 12.3 nM T64567 CJ4O2E 21806575 Ki = 3.8 nM T64567 CO2U7W 21855445 Ki = 5 nM T64567 CZ45AO 21878638 Ki = 226.9 nM T64567 C4XAO7 21879009 Ki = 98.5 nM T64567 CBS63Q 21879398 Ki = 171.1 nM T64567 C02IPY 21978067 Ki = 13.2 nM T64567 C6IZW0 22132896 Ki = 31 nM T64567 C9U4TE 22313850 Ki = 279 nM T64567 CX4Z1D 22315539 Ki = 20 nM T64567 C81ROV 22316829 Ki = 15 nM T64567 CPR25C 22706805 Ki = 920 nM T64567 C2D8ZL 23111570 Ki = 0.9 nM T64567 C2DOR4 23263451 Ki > 10000 nM T64567 C9KMP4 23275795 Ki = 0.89 nM T64567 CY6D4N 23644659 Ki = 3.6 nM T64567 CD5KT2 23644664 Ki = 213 nM T64567 C52YRI 23645366 Ki = 15 nM T64567 C3BSJ4 23645367 Ki = 8.7 nM T64567 CE50QI 23645368 Ki = 56 nM T64567 CNL51U 23645369 Ki = 3.2 nM T64567 CPRX73 23645370 Ki = 9 nM T64567 C9WT2E 23645682 Ki = 203 nM T64567 CU1OK9 23645683 Ki = 209 nM T64567 CLHE50 23645684 Ki = 85 nM T64567 C0UXY9 23646323 Ki = 103 nM T64567 C3QLX1 23646324 Ki = 420 nM T64567 CMX1A6 23646325 Ki = 114 nM T64567 C29HMI 23646326 Ki = 96 nM T64567 CCW81X 23647027 Ki = 72 nM T64567 CE20BX 23647028 Ki = 103 nM T64567 CNS87E 23661710 Ki = 22000 nM T64567 C8YRU5 23661711 Ki = 5050 nM T64567 CRZT32 23665339 Ki = 0.92 nM T64567 C7V6YP 23665706 Ki = 81.3 nM T64567 CXWP91 23666732 Ki = 4.5 nM T64567 C6W2BA 23668541 Ki = 678 nM T64567 CU08IW 23670409 Ki = 12.5 nM T64567 C1HCX5 23671974 Ki = 27.4 nM T64567 CDB01O 23674157 Ki = 6.8 nM T64567 CR7O3Q 23677931 Ki = 4.3 nM T64567 CKL59B 23679442 Ki = 8.1 nM T64567 CC93FA 23686905 Ki = 19.2 nM T64567 CZD6O0 23688497 Ki = 78.8 nM T64567 CE91KL 23691977 Ki = 322 nM T64567 CK2Q0I 23697126 Ki = 25.1 nM T64567 CPX0I4 24204718 Ki = 9.5 nM T64567 CF83JT 24204719 Ki = 39 nM T64567 CSWR58 24204720 Ki = 33 nM T64567 CIQ9L6 24204924 Ki = 18 nM T64567 CL2V5T 24204925 Ki = 13 nM T64567 C14RLU 24204932 Ki = 17 nM T64567 CN5ST6 24206002 Ki = 25 nM T64567 CPD4Z6 24206003 Ki = 25 nM T64567 C1Y2JB 24286289 Ki = 5.3 nM T64567 CKE1A3 24416843 Ki = 3.4 nM T64567 CA3Y8I 24588559 Ki = 240 nM T64567 CG98KI 24588612 Ki = 248 nM T64567 CK79DN 24588735 Ki = 197 nM T64567 CGHW54 24640576 Ki = 8 nM T64567 C01LHS 24640776 Ki = 16.8 nM T64567 CT8O2Z 24643222 Ki = 4.8 nM T64567 CB6WE3 24650532 Ki = 233 nM T64567 C1I9HZ 24692821 Ki = 159 nM T64567 CQG9O0 24816432 Ki = 11 nM T64567 CX10RQ 24823136 Ki = 120 nM T64567 CAS51H 24823137 Ki = 9.9 nM T64567 CXV0A1 24823299 Ki = 5 nM T64567 CK0D4U 24823300 Ki = 78.9 nM T64567 CU6VO3 24823301 Ki = 85 nM T64567 C8A9PE 24823302 Ki = 121 nM T64567 C5W7AC 24823303 Ki = 120 nM T64567 CZMT56 24823304 Ki = 110 nM T64567 CB9U5Z 24823476 Ki = 101 nM T64567 CXT1C5 24823477 Ki = 100 nM T64567 CBDO71 24823478 Ki = 134 nM T64567 CUT3V8 24823479 Ki = 120 nM T64567 C3UYV0 24823480 Ki = 130 nM T64567 CJQ3M4 24823631 Ki = 8.4 nM T64567 CPQN52 24823632 Ki = 5.4 nM T64567 CN75LK 24823633 Ki = 28 nM T64567 CNR3U7 24866945 IC50 > 10000 nM T64567 CQRZ10 24877657 Ki = 5.9 nM T64567 CCOG78 24944524 Ki = 18540 nM T64567 C62DIS 25048179 Ki = 301.2 nM T64567 COI25U 25131351 Ki = 165 nM T64567 CNMY17 25131685 Ki = 253 nM T64567 CB7V8Y 25147773 Ki = 3.3 nM T64567 C3KF1V 25178145 Ki = 12 nM T64567 C8PMK7 25178356 Ki = 26 nM T64567 C9HZG2 25181078 Ki = 3.8 nM T64567 CMYP34 25181079 Ki = 6.4 nM T64567 C7U1YC 25181080 Ki = 13 nM T64567 C85HLG 25181081 Ki = 13 nM T64567 C5T1NZ 25294048 Ki = 228.5 nM T64567 CRP6F5 25335375 Ki = 66 nM T64567 CPN2T5 25392418 Ki = 76.7 nM T64567 C1AOB3 25981084 Ki = 1.8 nM T64567 CP02LF 26365005 Ki = 6.5 nM T64567 C0RF4D 26470767 Ki = 201 nM T64567 CMUT78 26500397 Ki = 4.9 nM T64567 C5EC2T 26535209 Ki = 33.1 nM T64567 CLNR46 26598995 Ki = 188.9 nM T64567 CA9UZ7 26773685 Ki = 3.4 nM T64567 C8KQ5N 27868059 Ki = 69.1 nM T64567 CQSA29 27868075 Ki = 6.9 nM T64567 C7QB8M 27868953 Ki = 514 nM T64567 CWU2R0 27869227 Ki = 237 nM T64567 C46OQT 27869236 Ki = 462 nM T64567 C85HLF 27869237 Ki = 8.7 nM T64567 C5OWP7 27869350 Ki = 58.8 nM T64567 CF02EA 27869546 Ki = 39.6 nM T64567 C1G3XO 27869982 Ki = 69.3 nM T64567 C8ML3W 27870055 Ki = 24.5 nM T64567 CMK25I 27870443 Ki = 7.3 nM T64567 CQK4O6 27870796 Ki = 5.4 nM T64567 C2Z4FP 27870803 Ki = 53 nM T64567 C3RG8K 28846439 Ki = 10.7 nM T64567 C4EB0J 29034199 Ki = 2.4 nM T64567 CF8SA7 29559803 Ki = 2.2 nM T64567 CBPO08 34751720 Ki = 3121.2 nM T64567 CF3HA1 35871284 Ki = 20.1 nM T64567 CI0K1J 36865965 Ki = 3.1 nM T64567 C5IUO9 38154971 Ki = 219 nM T64567 CZE95V 38155699 Ki = 116 nM T64567 CSB4C7 38159448 Ki = 178 nM T64567 C4F7YT 40086402 Ki = 1570 nM T64567 C06EUO 40662472 Ki = 76.1 nM T64567 C1U4TL 41180562 Ki = 87 nM T64567 CH2P6W 41430216 Ki = 376 nM T64567 C5YBO2 41484755 Ki = 102 nM T64567 CUK13R 41874556 Ki = 22.1 nM T64567 C0J8DM 42597612 Ki = 4150 nM T64567 C8A5CF 42597613 Ki = 4190 nM T64567 C58ZUN 42597614 Ki = 4190 nM T64567 COG2A0 42597615 Ki = 4030 nM T64567 C1J9CQ 42597616 Ki = 3950 nM T64567 COG2I5 42598921 Ki = 4080 nM T64567 CDXS12 42598922 Ki = 4220 nM T64567 CP7UM8 42643988 Ki = 119000 nM T64567 C0IE3B 42644449 Ki = 9800 nM T64567 CT2C3D 42644450 Ki = 772000 nM T64567 CYJ0H4 43089860 Ki = 2.4 nM T64567 CXJY80 43235186 Ki = 2.6 nM T64567 C7EO2A 43329592 Ki = 3.5 nM T64567 CA0DX4 43342474 Ki = 7.4 nM T64567 C2HY4R 43342475 Ki = 2.4 nM T64567 CBK0M6 43342481 Ki = 1.3 nM T64567 C41VHR 43468983 Ki = 171 nM T64567 C82MRL 44144383 Ki = 6.4 nM T64567 CVJ5A1 44246262 Ki = 5.4 nM T64567 CZKG76 44246264 Ki = 3.5 nM T64567 C3E0CZ 44246268 Ki = 6.4 nM T64567 C0QZI4 44246269 Ki = 57 nM T64567 CZL01D 44246271 Ki = 63 nM T64567 C6V9WT 44309709 Ki = 39 nM T64567 CYUE74 44309710 Ki = 44 nM T64567 CERI42 44309802 Ki = 34 nM T64567 CLBU37 44310092 Ki = 32 nM T64567 CW0S8U 44311169 Ki = 24 nM T64567 C76HLZ 44314854 Ki = 12 nM T64567 C91HDR 44315566 Ki = 43.1 nM T64567 CAPN36 44367390 Ki > 1000 nM T64567 CS4P3F 44367405 Ki = 13 nM T64567 CD98KU 44367410 Ki = 76 nM T64567 CF8J7B 44367431 Ki = 65 nM T64567 CE18VJ 44367432 Ki > 1000 nM T64567 CT0R9B 44367463 Ki = 17 nM T64567 CI8PB1 44391626 Ki = 9.6 nM T64567 C68BRH 44391633 Ki = 70.8 nM T64567 C6BUC8 44391791 Ki = 163 nM T64567 CWR3F1 44391802 Ki = 235 nM T64567 CM6F7X 44391805 Ki = 35 nM T64567 C93OPV 44391820 Ki = 67 nM T64567 CDH40E 44391824 Ki = 31 nM T64567 CUK9X4 44391833 Ki = 33 nM T64567 COTH27 44391859 Ki = 90 nM T64567 C5ZA9R 44395106 Ki = 1.1 nM T64567 C4OR5F 44395107 Ki = 150 nM T64567 C9J2ME 44395133 Ki = 138 nM T64567 C9MLB4 44395134 Ki = 142 nM T64567 CI3O9B 44395149 Ki = 153 nM T64567 CO8J7I 44395150 Ki = 1.3 nM T64567 CPB8W7 44395163 Ki = 124 nM T64567 C8EK1N 44395173 Ki = 360 nM T64567 CQ54DL 44395174 Ki = 549 nM T64567 CWUP51 44395202 Ki = 0.12 nM T64567 CIWO28 44395243 Ki = 155 nM T64567 CYR62U 44395244 Ki = 162 nM T64567 CUW0D8 44395258 Ki = 12 nM T64567 C6H1QR 44395691 Ki = 18 nM T64567 CWN75T 44395718 Ki = 20 nM T64567 CR81IG 44395747 Ki = 18 nM T64567 CYS09N 44395778 Ki = 23 nM T64567 CX9RC2 44395866 Ki = 3.2 nM T64567 CN7A1U 44395892 Ki = 19 nM T64567 C90XMR 44395897 Ki = 10 nM T64567 CVC7K9 44395919 Ki = 3 nM T64567 CA65VH 44398374 Ki = 38 nM T64567 C7T8XG 44399285 Ki = 16 nM T64567 CNSR28 44399286 Ki = 6.3 nM T64567 C8NOW9 44399298 Ki = 2.5 nM T64567 C89LNG 44399317 Ki = 1.5 nM T64567 CT3V7P 44399318 Ki = 386 nM T64567 CCD34Q 44399321 Ki = 1.5 nM T64567 C67HFO 44399335 Ki = 56 nM T64567 CQJZ93 44399338 Ki = 81 nM T64567 C0KFU7 44399339 Ki = 84 nM T64567 CH6GT7 44399340 Ki = 7.3 nM T64567 CG0Z9A 44399346 Ki = 210 nM T64567 C8EQG2 44399347 Ki = 113 nM T64567 C5GJ3N 44399351 Ki = 1.4 nM T64567 CNTM52 44399371 Ki = 13 nM T64567 C3QZR6 44399393 Ki = 7.5 nM T64567 C7BHR6 44399404 Ki = 1.3 nM T64567 C7LCX4 44399427 Ki = 12.6 nM T64567 C48MQR 44399437 Ki = 185 nM T64567 CCZG27 44399440 Ki = 1 nM T64567 C72HQK 44399449 Ki = 9.3 nM T64567 CGEX61 44399456 Ki = 197 nM T64567 CU1B9T 44399459 Ki = 174 nM T64567 CV9EU2 44399460 Ki = 287 nM T64567 CQCB53 44399461 Ki = 274 nM T64567 CZ4DF9 44399462 Ki = 1 nM T64567 CZ3YC5 44399486 Ki = 2.9 nM T64567 CVK1X8 44399489 Ki = 18 nM T64567 CUK37Q 44399499 Ki = 5.9 nM T64567 CVP43X 44399501 Ki = 10.5 nM T64567 CRM73I 44399515 Ki = 1.4 nM T64567 CK6G2Y 44399516 Ki = 423 nM T64567 C4UEG1 44399517 Ki = 640 nM T64567 CL6F3X 44399532 Ki = 125 nM T64567 CU7BK9 44399535 Ki = 1.2 nM T64567 CX6B8J 44399541 Ki = 78 nM T64567 CMFY95 44399542 Ki = 13.7 nM T64567 C8B9NK 44399547 Ki = 254 nM T64567 CT57KL 44399549 Ki = 1.2 nM T64567 CB0R2P 44399570 Ki = 204 nM T64567 CD5MJ6 44399571 Ki = 1.7 nM T64567 C3EBD7 44399585 Ki = 80 nM T64567 C0RT3E 44399598 Ki = 84 nM T64567 CPKG57 44399624 Ki = 7.6 nM T64567 CI5Y0H 44399639 Ki = 81 nM T64567 C2T7MB 44399654 Ki = 81 nM T64567 CU3DY1 44399655 Ki = 80 nM T64567 C4AD1R 44399664 Ki = 53 nM T64567 CR95YM 44399687 Ki = 89 nM T64567 CGC2M5 44399695 Ki = 42 nM T64567 C3W9CF 44399734 Ki = 10.1 nM T64567 CUXT35 44401673 Ki = 5.4 nM T64567 C4AD6B 44401689 Ki = 5.6 nM T64567 C1A5NV 44401728 Ki = 5 nM T64567 CWJ08B 44401743 Ki = 256000 nM T64567 C83EIL 44401769 Ki = 6.7 nM T64567 C2HDZ6 44401810 Ki = 192000 nM T64567 CJ86PU 44401826 Ki = 6.7 nM T64567 C0F1VY 44401832 Ki = 271000 nM T64567 CQ02ZD 44401833 Ki = 322000 nM T64567 C5PR9E 44401857 Ki = 4.8 nM T64567 C7NM9T 44401871 Ki = 242000 nM T64567 CYQF42 44401889 Ki = 4.8 nM T64567 CIN38J 44401926 Ki = 320000 nM T64567 C75WFG 44401951 Ki = 315000 nM T64567 CX1LH3 44401952 Ki = 6.4 nM T64567 CIO61G 44401975 Ki = 312000 nM T64567 C9M0ID 44401978 Ki = 296000 nM T64567 C34PLI 44402062 Ki = 60400 nM T64567 CF6X9Y 44402148 Ki = 6.1 nM T64567 C28JBO 44402274 Ki = 5.2 nM T64567 CGPF38 44402275 Ki = 4.6 nM T64567 CT6UF5 44402709 Ki = 32 nM T64567 C5FC0Y 44402716 Ki > 1000 nM T64567 C8N0GW 44402748 Ki = 45 nM T64567 C9AJ7Z 44402772 Ki = 26 nM T64567 CR72VG 44402825 Ki = 30 nM T64567 C5LU4G 44403258 Ki = 13 nM T64567 C6OS3R 44403265 Ki = 13 nM T64567 CI18FK 44403266 Ki = 362 nM T64567 CR2Z7F 44403267 Ki = 76 nM T64567 C0W6BQ 44403268 Ki > 1000 nM T64567 C8QXA6 44403278 Ki > 1000 nM T64567 CSN79Y 44403312 Ki = 37 nM T64567 CW93DL 44405187 Ki = 240 nM T64567 CSXF07 44405190 Ki = 195 nM T64567 CVJ5T9 44416166 Ki = 40.9 nM T64567 CZT1U9 44416167 Ki > 10000 nM T64567 CQ36IP 44416168 Ki = 56 nM T64567 CS49FE 44416185 Ki = 5440 nM T64567 CEH5P1 44416186 Ki = 4995 nM T64567 C8C4IJ 44416203 Ki > 10000 nM T64567 CE6N7Q 44416215 Ki > 10000 nM T64567 CY9VT1 44416239 Ki = 113 nM T64567 CI01QM 44416240 Ki = 139 nM T64567 CX8ZQ9 44416241 Ki > 10000 nM T64567 CRX27F 44416256 Ki = 780 nM T64567 C68YLB 44416306 Ki = 1613 nM T64567 C5ROE2 44416307 Ki = 1440 nM T64567 C47OTU 44416317 Ki = 3415 nM T64567 CE4M9P 44416378 Ki = 766 nM T64567 CE03DL 44416379 Ki > 10000 nM T64567 C67IEM 44420782 Ki = 84 nM T64567 CY49HT 44423674 Ki = 9000 nM T64567 CHI5G1 44423675 Ki = 7500 nM T64567 CFC3M6 44423676 Ki = 9300 nM T64567 CO24JF 44423677 Ki = 9500 nM T64567 C7F9DB 44423678 Ki = 7400 nM T64567 CJ6GW5 44423679 Ki = 7800 nM T64567 CUKM29 44423680 Ki = 8700 nM T64567 C3R0FS 44423681 Ki = 9300 nM T64567 C14DBJ 44423682 Ki = 9200 nM T64567 CP3OY8 44428369 Ki = 34.1 nM T64567 CM3J0U 44430517 Ki = 10 nM T64567 C9LT7Y 44430518 Ki = 82 nM T64567 C1VTB6 44430520 Ki = 4500 nM T64567 C2L5MB 44430521 Ki = 134 nM T64567 CVEO17 44430523 Ki = 11 nM T64567 C8MFL1 44430524 Ki = 76 nM T64567 CW8DJ9 44435841 Ki = 9300 nM T64567 CQ4RC2 44435843 Ki = 23000 nM T64567 C9RYT1 44435845 Ki = 7130 nM T64567 CHDA78 44435846 Ki = 24000 nM T64567 C1G7HL 44435848 Ki = 29000 nM T64567 CW3M0X 44435849 Ki = 118220 nM T64567 CA4ZH8 44435850 Ki = 10100 nM T64567 CW73VG 44435851 Ki = 7530 nM T64567 C3D6AL 44435853 Ki = 24000 nM T64567 C6X5NI 44435855 Ki = 10000 nM T64567 COUY42 44435856 Ki = 3350 nM T64567 C1LM4Y 44435857 Ki = 7440 nM T64567 CU72AI 44435858 Ki = 148900 nM T64567 C5AMH4 44435861 Ki = 20000 nM T64567 C38GXC 44435862 Ki = 8550 nM T64567 C1AOX2 44435863 Ki = 6850 nM T64567 CFBT23 44435864 Ki = 7540 nM T64567 C37DRO 44435865 Ki = 8430 nM T64567 CT3S5B 44435866 Ki = 5750 nM T64567 C3PTQ7 44435867 Ki = 8830 nM T64567 C74ECN 44448778 Ki = 35 nM T64567 CX50NI 44448882 Ki = 41 nM T64567 CNRW48 44448977 Ki = 41 nM T64567 CUWK18 44449006 Ki = 7 nM T64567 CB9KU0 44449032 Ki = 30 nM T64567 CSFE58 44449055 Ki = 220 nM T64567 CV31AN 44449057 Ki = 14 nM T64567 C7PU2N 44449080 Ki = 22 nM T64567 CLIV87 44449082 Ki = 39 nM T64567 C48XSU 44449083 Ki = 132 nM T64567 C8P4EB 44459430 Ki = 41 nM T64567 CNW10Y 44459431 Ki = 23 nM T64567 CQUC34 44520900 Ki = 11 nM T64567 CHCT21 44542292 Ki = 7.3 nM T64567 CG61YX 44542293 Ki = 7.1 nM T64567 CL8AQ5 44542294 Ki = 6.3 nM T64567 CF2RX4 44542600 Ki = 7.9 nM T64567 C5MZ3O 44542742 Ki = 6.5 nM T64567 CI9VZ6 44542743 Ki = 7.4 nM T64567 C18XNW 44564181 Ki = 1840 nM T64567 CQIJ49 44564248 Ki = 90 nM T64567 CR8V7Q 44564282 Ki = 10 nM T64567 C64APD 44574189 Ki = 8440 nM T64567 CV5XS1 44574190 Ki = 8200 nM T64567 CE0ZS5 44574217 Ki = 7540 nM T64567 C3OYU7 44574218 Ki = 4980 nM T64567 CHJV65 44574219 Ki = 5590 nM T64567 C4FI0H 44574220 Ki = 6750 nM T64567 CM9E2T 44574221 Ki = 6450 nM T64567 C5MCT7 44574248 Ki = 480 nM T64567 CZB19D 44574249 Ki = 8130 nM T64567 C48VUR 44574250 Ki = 6780 nM T64567 CH03WX 44577410 Ki = 76 nM T64567 CCH53K 44577411 Ki = 23 nM T64567 CKT85S 44577800 Ki = 25.9 nM T64567 C3DU8S 44577801 Ki = 22.4 nM T64567 CCW3S1 44578981 Ki = 113 nM T64567 CU7Y8T 44578982 Ki = 91 nM T64567 C86YLD 44579460 Ki = 59 nM T64567 CD4WO8 44579535 Ki = 14 nM T64567 CF0KQ8 44581932 Ki = 38 nM T64567 CM2L4W 44591861 Ki = 8.1 nM T64567 CSU20V 44591862 Ki = 101 nM T64567 CF9MS6 44591908 Ki = 101 nM T64567 CQ40FB 44592373 Ki = 8.6 nM T64567 C15THP 44592446 Ki = 9.9 nM T64567 CDB3X7 44592447 Ki = 9.3 nM T64567 C2J3ER 44592448 Ki = 8.6 nM T64567 CUXJ39 44592449 Ki = 7.7 nM T64567 CTI2C1 44592450 Ki = 7.5 nM T64567 COS6N0 44592512 Ki = 257 nM T64567 CASL51 44592513 Ki = 9.8 nM T64567 CXL68J 44592514 Ki = 9.5 nM T64567 COL03N 44592515 Ki = 6.1 nM T64567 CHMW14 44592516 Ki = 8 nM T64567 COX6D8 45028566 Ki = 13.5 nM T64567 CF2WL9 45028890 Ki = 68 nM T64567 C4MO3S 45028891 Ki = 6.9 nM T64567 C80CDA 45028892 Ki = 18.3 nM T64567 C6YHW4 45028893 Ki = 5.2 nM T64567 C16ILW 45028894 Ki = 5.8 nM T64567 CA07CZ 45268031 Ki = 840 nM T64567 CMUX83 45268595 Ki = 8.8 nM T64567 C23MVW 45269009 IC50 = 54500 nM T64567 C0RG8K 45269749 Ki = 8200 nM T64567 CKFY69 45270284 Ki = 220 nM T64567 C6E7XJ 45484068 Ki = 3910 nM T64567 CGI25L 45484069 Ki = 4090 nM T64567 CVG6K1 45484072 Ki = 4050 nM T64567 CV5RQ3 45484187 Ki = 54.5 nM T64567 CTG20B 45485271 Ki = 3000 nM T64567 CK4U0V 45485283 Ki = 8700 nM T64567 C5GZ1B 46197458 Ki = 105 nM T64567 C3Z7OL 46197569 Ki = 91 nM T64567 CUQF42 46197571 Ki = 100 nM T64567 C4C7XG 46197572 Ki = 84 nM T64567 CLBG91 46197677 Ki = 79 nM T64567 C9GC5Q 46197678 Ki = 89 nM T64567 C16XCV 46197680 Ki = 102 nM T64567 C3JW1R 46197790 Ki = 88 nM T64567 CD49XQ 46197791 Ki = 95 nM T64567 C4H9TD 46197792 Ki = 99 nM T64567 C0W1GZ 46197794 Ki = 106 nM T64567 CUO20Q 46197893 Ki = 98 nM T64567 CN7KI3 46197894 Ki = 97 nM T64567 CD74LO 46197895 Ki = 107 nM T64567 CZ93SW 46197897 Ki = 97 nM T64567 CNQZ73 46197997 Ki = 94 nM T64567 CCAX25 46197998 Ki = 95 nM T64567 CQ3R2U 46197999 Ki = 96 nM T64567 CGM42H 46198111 Ki = 97 nM T64567 C0DKY8 46198112 Ki = 93 nM T64567 CBWN61 46198113 Ki = 84 nM T64567 C0AF1L 46198114 Ki = 100 nM T64567 C1KWB5 46198220 Ki = 100 nM T64567 CEV26X 46198221 Ki = 81 nM T64567 C1ALN3 46201612 Ki = 80 nM T64567 C25FBC 46567082 Ki = 14.6 nM T64567 CQN8K4 46635132 Ki = 46 nM T64567 CA4FJ2 46703925 Ki = 4.6 nM T64567 C2WB4C 46703927 Ki = 9.6 nM T64567 CO2IU4 46704079 Ki = 7.5 nM T64567 CB85EQ 46704080 Ki = 7.2 nM T64567 CAE9Z3 46704081 Ki = 5.8 nM T64567 CD5V6T 46704082 Ki = 16.1 nM T64567 C8MR0H 46847340 IC50 = 7000 nM T64567 CRS8J6 46860267 Ki = 73.3 nM T64567 C2RA7G 46861342 Ki = 49.1 nM T64567 C2S4YC 46866644 IC50 = 7000 nM T64567 C7QR8Y 46866645 IC50 = 6800 nM T64567 CUH07J 46866646 IC50 = 6100 nM T64567 C8GK4C 46866647 IC50 = 6300 nM T64567 C7CQ6I 46871755 Ki = 8.5 nM T64567 CNEO10 46871889 Ki = 130 nM T64567 C7UKN2 46884029 Ki = 102 nM T64567 C1DCM9 46884093 Ki = 89 nM T64567 C4ALG9 46884132 Ki = 97 nM T64567 CTRY21 46884169 Ki = 90 nM T64567 CBM20W 46884215 Ki = 95 nM T64567 CR61DW 46884254 Ki = 96 nM T64567 C0AN1G 46890958 Ki = 3.4 nM T64567 C08WJF 46890959 Ki = 3.5 nM T64567 C9UK8S 46891017 Ki = 4.1 nM T64567 C2KT4I 46891018 Ki > 1000 nM T64567 C93AIR 46899573 Ki = 117000 nM T64567 C4GZ6A 46907387 Ki = 7.7 nM T64567 CJ0R2O 46911381 Ki = 49.5 nM T64567 C6YK2E 46913624 Ki = 2.5 nM T64567 CAF1K0 46913625 Ki > 1000 nM T64567 CO60NB 46918149 Ki > 1000 nM T64567 C9T3WF 46933594 Ki = 64 nM T64567 C1WE2D 46933744 Ki = 11.8 nM T64567 CUHI56 46933745 Ki = 9.7 nM T64567 C27DFQ 46933746 Ki = 8.6 nM T64567 CSQG87 46933747 Ki = 10.1 nM T64567 C08BKN 46933748 Ki = 11.9 nM T64567 C54PRX 46933749 Ki = 118 nM T64567 CP62AV 46933896 Ki = 96 nM T64567 C03FQY 46943413 Ki = 65.7 nM T64567 C31ZQL 49843495 Ki = 10 nM T64567 CQJX35 49843496 Ki = 11 nM T64567 CCOB94 49929067 Ki = 2.5 nM T64567 CY45IU 49957432 IC50 = 0.3 nM T64567 C5Z2QA 50741845 Ki = 89 nM T64567 CVC35K 50899076 IC50 = 9000 nM T64567 CR3I2H 50899077 IC50 = 8800 nM T64567 CEHP41 50909907 Ki = 0.9 nM T64567 CB4O0Y 50909908 Ki = 0.5 nM T64567 C1QBZ3 50942416 Ki = 0.8 nM T64567 C62ZDQ 51035422 Ki = 0.75 nM T64567 CW0CJ2 51035423 Ki = 8.2 nM T64567 C5CR2F 51039206 Ki = 7.8 nM T64567 C3SH7R 51039207 Ki = 8.4 nM T64567 CS5ZR3 51039209 Ki = 9 nM T64567 C8TR3Z 51047320 Ki = 2.6 nM T64567 CHK5G9 51059586 Ki > 50000 nM T64567 C8XGV5 51349458 Ki = 73 nM T64567 C4S5NC 51349459 Ki = 77 nM T64567 CZH4T2 51349599 Ki = 86 nM T64567 CK3U6Q 51349600 Ki = 75 nM T64567 CDF2V8 51349601 Ki = 631 nM T64567 CG26DK 51349604 Ki = 497 nM T64567 CUP39M 51355749 Ki = 47.1 nM T64567 CJ1M5T 51355750 Ki = 6 nM T64567 CBL9U1 51356010 Ki = 65.7 nM T64567 CLG43P 51669707 IC50 = 7140 nM T64567 C1FM4S 52940811 Ki = 111 nM T64567 CE15GD 52941031 Ki = 89 nM T64567 CE7WD6 52942084 Ki = 83 nM T64567 CRMY05 52942168 Ki = 200 nM T64567 C7OA0E 52942246 Ki = 101 nM T64567 C4O3HF 52942279 Ki = 3.7 nM T64567 C2OQL5 52942476 Ki = 63.9 nM T64567 C0R5HD 52943223 Ki = 68 nM T64567 CCNT92 52943270 Ki = 147 nM T64567 CXMY91 52943276 Ki = 22 nM T64567 CC67HN 52943455 Ki = 135 nM T64567 C50ELG 52943614 Ki > 100000 nM T64567 C7HU5Q 52944525 Ki = 133 nM T64567 CB4UY1 52944603 Ki = 242 nM T64567 C3G6WM 52944864 Ki > 100000 nM T64567 C20FAL 52945268 Ki = 187 nM T64567 C3MLZ1 52945326 Ki = 207 nM T64567 CBGN39 52945721 Ki = 137 nM T64567 CCV6U5 52945740 Ki = 167 nM T64567 CX28EM 52945837 Ki = 4.7 nM T64567 C6ZCQ2 52947045 Ki = 125 nM T64567 CRVI93 52948047 Ki > 100000 nM T64567 CDNI78 52948211 Ki = 30 nM T64567 CAW78K 52948213 Ki = 126 nM T64567 CA59GT 52948974 Ki = 198 nM T64567 C14WUN 52949402 Ki = 153 nM T64567 CW92IL 52949544 Ki = 131 nM T64567 CLK0S1 52950139 Ki > 1000 nM T64567 CPGW70 53245686 Ki = 235 nM T64567 CCW69Q 53308637 Ki = 96 nM T64567 CKRO12 53321135 Ki = 53 nM T64567 CTF92V 53322463 Ki = 8.6 nM T64567 C8Z2IL 53324362 Ki = 62 nM T64567 CK4ZG3 53342705 Ki = 3.788 nM T64567 CHF62Q 53361485 IC50 = 347 nM T64567 CJ3F4R 53361486 IC50 = 6131 nM T64567 C08REF 53364160 Ki = 13 nM T64567 C32UEX 53364161 Ki = 16 nM T64567 CHWX25 53364162 Ki = 5 nM T64567 C3OUP0 53364163 Ki = 5 nM T64567 C58YMC 53371608 Ki = 12 nM T64567 C0NUM6 53386724 Ki = 18.5 nM T64567 C54FGU 53386866 Ki = 24 nM T64567 CRI54V 53386867 Ki = 10.2 nM T64567 CUX7S4 53386868 Ki = 19.4 nM T64567 CSA60L 53389267 Ki = 115 nM T64567 C8VXD9 53389268 Ki = 1.5 nM T64567 CV40HR 53426278 Ki = 3.6 nM T64567 C6T5RC 53483944 Ki = 6.5 nM T64567 CM5KX6 53483945 Ki = 1.7 nM T64567 C3M4EL 53483958 Ki = 8450 nM T64567 CCFP92 53516400 Ki = 6.5 nM T64567 CY2MI0 54077127 Ki = 188 nM T64567 CB6W4D 54577841 Ki = 31.8 nM T64567 CI83DC 54578707 Ki = 7.7 nM T64567 CHCT45 54580732 Ki = 25 nM T64567 CYB47X 54581736 Ki = 11 nM T64567 CW2KI4 54582723 Ki = 10 nM T64567 CWK6B0 54582724 Ki = 85 nM T64567 CBS8R1 54584666 Ki = 177 nM T64567 CJ3UE2 54584667 Ki = 93 nM T64567 CO0BD9 54585508 Ki = 83 nM T64567 C0A5OZ 54612935 Ki = 12.6 nM T64567 C6SM5T 54613427 Ki = 76 nM T64567 C6X7QG 54613732 Ki = 2.4 nM T64567 CKB0G9 54669765 Ki = 6.2 nM T64567 CS8IV7 54669781 Ki = 6.5 nM T64567 C0PJ1K 54677403 Ki = 35.9 nM T64567 CAS91K 54682930 Ki = 410 nM T64567 CQ3XK0 54758050 Ki = 95 nM T64567 C5ON9E 54758136 Ki = 71 nM T64567 C0K2LN 54758137 Ki = 97 nM T64567 C5Q9XC 54758138 Ki = 99.6 nM T64567 CLT0W2 54758232 Ki = 61.9 nM T64567 C5V4GI 54758233 Ki = 7.3 nM T64567 C98JVL 54758234 Ki = 61 nM T64567 CXBF42 54758235 Ki = 89 nM T64567 C4EL5V 54758236 Ki = 68 nM T64567 CU19DH 54758322 Ki = 71.2 nM T64567 CE53AN 54758323 Ki = 72 nM T64567 CK3Q0O 54758324 Ki = 91 nM T64567 CE2O3A 54768697 Ki = 8.7 nM T64567 C5SB4M 54768698 Ki = 10.2 nM T64567 CBNP25 54768699 Ki = 9 nM T64567 C9Z4RJ 54772055 Ki = 7.6 nM T64567 CB3EC8 54772057 Ki = 7.4 nM T64567 CE6LD4 54772059 Ki = 10.1 nM T64567 CD5P1I 54772061 Ki = 9 nM T64567 C3RQX8 54940826 Ki = 274 nM T64567 CK89GH 56659335 Ki = 9.4 nM T64567 C05JRQ 56659336 Ki = 8.5 nM T64567 CEC29W 56659337 Ki = 8.4 nM T64567 C2TW1F 56659553 Ki = 9.3 nM T64567 CO9SW8 56659554 Ki = 91 nM T64567 CVRM21 56659555 Ki = 8.6 nM T64567 CJ43WP 56659826 Ki = 900 nM T64567 CZ4HI1 56662794 Ki = 8.9 nM T64567 CD8SR3 56662795 Ki = 34.8 nM T64567 CF0J6I 56663002 Ki = 9.5 nM T64567 CH0MV2 56663442 Ki = 69 nM T64567 CM07OK 56663443 Ki = 1 nM T64567 CVM8W4 56666268 Ki = 8.4 nM T64567 C89SEG 56666269 Ki = 34.1 nM T64567 C36TYE 56666270 Ki = 9 nM T64567 CD5OZ4 56666482 Ki = 9.6 nM T64567 CI93KS 56666719 Ki = 900 nM T64567 CR9F8U 56670316 Ki = 1.6 nM T64567 CF1J7H 56670317 Ki = 8600 nM T64567 CWNF20 56673403 Ki = 89 nM T64567 CT29KP 56673404 Ki = 92 nM T64567 C7DU3M 56673405 Ki = 9 nM T64567 CHV04E 56673655 Ki = 5.3 nM T64567 C4YI1B 56673656 Ki = 900 nM T64567 CKL09N 56673817 Ki = 1.1 nM T64567 CI2R9B 56676517 Ki = 8.9 nM T64567 C9X7VM 56676518 Ki = 0.96 nM T64567 CF86WB 56676713 Ki = 7.7 nM T64567 CDH07V 56677155 Ki = 68 nM T64567 CR7D6S 56677156 Ki = 6370 nM T64567 C2U1VF 56679839 Ki = 9.2 nM T64567 CS81JH 56680034 Ki = 9.5 nM T64567 C02WBE 56680461 Ki = 5.8 nM T64567 CEZ3F5 56683163 Ki = 113 nM T64567 C4LB1M 56683164 Ki = 95 nM T64567 CZS9V5 56683165 Ki = 91 nM T64567 C8V1PA 56683626 Ki = 5 nM T64567 CXL7Q1 56683627 Ki = 3140 nM T64567 CIJ9V0 56684131 Ki = 3250 nM T64567 C6IAC4 56689569 Ki = 8190 nM T64567 CTWZ62 56836370 Ki = 6.3 nM T64567 C49PBJ 56836371 Ki = 7.6 nM T64567 CK7Y8J 56836443 Ki = 154 nM T64567 CY7Z1A 56836444 Ki = 349 nM T64567 CV0ST7 56836445 Ki = 7.4 nM T64567 C0O3UI 56836446 Ki = 8.7 nM T64567 C0PKB5 56836447 Ki = 9.6 nM T64567 CZ9F7P 56836511 Ki = 6.1 nM T64567 COY29V 56836512 Ki = 8.9 nM T64567 C7PWG1 56836513 Ki = 8.2 nM T64567 C4CF8M 56836514 Ki = 8.4 nM T64567 C4IRK8 56836515 Ki = 6.3 nM T64567 CH52DA 56921864 Ki = 2410 nM T64567 C0Z8WY 56925533 Ki = 820 nM T64567 CTFL92 56928044 Ki = 18.3 nM T64567 CC3Q9S 56928516 Ki = 6 nM T64567 CO18AP 57011620 Ki = 8.5 nM T64567 C4VGE9 57047254 Ki = 6.9 nM T64567 CNG76Q 57326130 Ki = 29.1 nM T64567 C81YCD 57326131 Ki = 22.1 nM T64567 C4TV1U 57326132 Ki = 4.6 nM T64567 CHL0B3 57326133 Ki = 4.5 nM T64567 C5Z4SW 57326134 Ki = 27.4 nM T64567 CFU62Y 57326227 Ki = 3.6 nM T64567 C97HYX 57326228 Ki = 4.3 nM T64567 CS4I5T 57326229 Ki = 4.1 nM T64567 CP7YR5 57345662 Ki = 16 nM T64567 C0S2YZ 57383964 Ki = 8.4 nM T64567 C97GHV 57383965 Ki = 2.1 nM T64567 CXW5D3 57384052 Ki = 800 nM T64567 C4XF9A 57384114 Ki = 7.4 nM T64567 CS76WU 57384115 Ki = 8.8 nM T64567 C0UBL5 57384116 Ki = 112 nM T64567 C16AGY 57384117 Ki = 121 nM T64567 CVWK43 57386884 Ki = 850 nM T64567 CR3C7D 57386885 Ki = 860 nM T64567 C9CX4B 57386886 Ki = 960 nM T64567 CZOD69 57386887 Ki = 800 nM T64567 CZN72E 57386888 Ki = 3040 nM T64567 C9JU0H 57386889 Ki = 3260 nM T64567 CQ0I4V 57386890 Ki = 530 nM T64567 C8Z0DJ 57387135 Ki = 680 nM T64567 C1HZS5 57387136 Ki = 610 nM T64567 C7EN6Z 57387137 Ki = 970 nM T64567 C87ASQ 57387395 Ki = 41600 nM T64567 CQW5T3 57387397 Ki = 830 nM T64567 CT3B0Z 57387636 Ki = 3230 nM T64567 CV4C7B 57390570 Ki = 21.8 nM T64567 CS5O2D 57390571 Ki = 7.5 nM T64567 C14VNC 57390572 Ki = 5 nM T64567 C09GQI 57392249 Ki = 6.9 nM T64567 CY81SU 57392250 Ki = 3.3 nM T64567 CMEV16 57392251 Ki = 122 nM T64567 C94YIX 57392252 Ki = 282 nM T64567 CDP3C2 57392352 Ki = 16 nM T64567 CM7S3H 57394009 Ki = 8.7 nM T64567 CHAF57 57394010 Ki = 9.1 nM T64567 CV7K9Y 57394771 Ki = 7 nM T64567 CM4SL9 57394772 Ki = 258 nM T64567 C1M0LS 57394809 Ki = 680 nM T64567 CJ5XK2 57395770 Ki = 451 nM T64567 CV6QX4 57395771 Ki = 433 nM T64567 CP9D5B 57395861 Ki = 60.7 nM T64567 CHG91B 57396529 Ki = 2.8 nM T64567 C9H4VS 57396530 Ki = 113 nM T64567 C6XD2O 57397549 Ki = 7.5 nM T64567 C64VIW 57397550 Ki = 8.9 nM T64567 CR30XN 57397648 Ki = 7 nM T64567 CRIU35 57398318 Ki = 115 nM T64567 CN6TU2 57398319 Ki = 8.9 nM T64567 C97OJM 57399231 Ki = 7.4 nM T64567 C7XAZ3 57399232 Ki = 362 nM T64567 CK24NA 57399233 Ki = 8.7 nM T64567 CQD65L 57401080 Ki = 31 nM T64567 C1SK7F 57401081 Ki = 12 nM T64567 CG3X4V 57401764 Ki = 8.3 nM T64567 C4V5KY 57402747 Ki = 7.3 nM T64567 CRU53E 57402748 Ki = 5.8 nM T64567 C52TUM 57402749 Ki = 7.5 nM T64567 CQ9ZG2 57402750 Ki = 7.3 nM T64567 CI3L9R 57402843 Ki = 78 nM T64567 CW10QX 57402844 Ki = 18 nM T64567 C80WTZ 57403496 Ki = 6.9 nM T64567 CDIM87 57403497 Ki = 8.4 nM T64567 C76ZDS 57404539 Ki = 7.2 nM T64567 CKID78 57411990 Ki = 4.3 nM T64567 C4ZYF3 57411991 Ki = 4.2 nM T64567 CDG6R4 57411992 Ki = 7.1 nM T64567 CKPS17 57411993 Ki = 5.2 nM T64567 CV13LT 57411994 Ki = 49 nM T64567 CW1TU4 57412422 Ki = 8.1 nM T64567 CT4BV9 57412423 Ki = 8.3 nM T64567 C31NWX 57412424 Ki = 41.7 nM T64567 CD86ER 57412425 Ki = 7.2 nM T64567 CB94YU 57412426 Ki = 16.1 nM T64567 C2K8YJ 57412507 Ki = 15.4 nM T64567 CSF4V6 57412508 Ki = 9.2 nM T64567 CHAO86 57412509 Ki = 9.2 nM T64567 C3U6TH 57412510 Ki = 68.3 nM T64567 C40LOS 57412511 Ki = 6.5 nM T64567 CZ47VT 57412512 Ki = 52.1 nM T64567 C28WRD 57412600 Ki = 6.5 nM T64567 C2XPG5 57413583 Ki = 7.8 nM T64567 CM2AY7 57413584 Ki = 7.9 nM T64567 C5JDQ1 57413825 Ki = 70 nM T64567 C5M4CN 57413826 Ki = 7.3 nM T64567 C3D7KS 57413827 Ki = 7.9 nM T64567 CJO26X 57413828 Ki = 8 nM T64567 CA4CD7 57413968 Ki = 20.4 nM T64567 CQ1ZK6 57519697 Ki = 64 nM T64567 CG3W0D 58404071 Ki = 400 nM T64567 C01TQW 59079460 Ki = 9.6 nM T64567 CF1NG0 60155028 Ki = 3.52 nM T64567 C0PRW7 60155029 Ki = 3.554 nM T64567 CNX97Q 60155030 Ki = 3.457 nM T64567 CR0Z7W 60155031 Ki = 3.202 nM T64567 CI2WL7 60155120 Ki = 3.855 nM T64567 CM57BF 60155121 Ki = 3.378 nM T64567 C5VF9X 60155122 Ki = 3.855 nM T64567 C2U8VH 60155123 Ki = 3.679 nM T64567 CNR53M 60155124 Ki = 14 nM T64567 CYQM98 60201413 Ki = 65 nM T64567 CGWU14 60201414 Ki = 611 nM T64567 C6TP2W 60201415 Ki = 27 nM T64567 C1JVP9 60201416 Ki = 35 nM T64567 CQZN79 60201417 Ki = 65 nM T64567 CVU0B4 60201577 Ki = 52 nM T64567 CS3N6M 60201578 Ki = 0.4 nM T64567 CB45GM 60201579 Ki = 4.5 nM T64567 C9V6EY 60446869 Ki = 3972 nM T64567 C1CVG9 61580845 Ki = 3.9 nM T64567 C9UD2V 62141270 Ki = 1398 nM T64567 CZ4BQ6 66571808 Ki = 8.2 nM T64567 CGB46T 66571809 Ki = 9.7 nM T64567 CT0S3A 66572208 Ki = 22.1 nM T64567 CGF3W6 66586679 Ki = 900 nM T64567 CN84CU 66586879 Ki = 810 nM T64567 CAD3V2 67662627 Ki = 31 nM T64567 C54HCL 68341722 Ki = 112.9 nM T64567 C4MB5P 68602550 Ki = 392 nM T64567 CA7F0J 68819643 Ki = 22 nM T64567 CV6PY2 68833705 Ki = 20.1 nM T64567 C23JZS 70037678 Ki = 24.7 nM T64567 C6RVC3 70202738 Ki = 9 nM T64567 CDO92J 70681983 Ki = 3.429 nM T64567 CHC54M 70681984 Ki = 3.429 nM T64567 C1FY3K 70681985 Ki = 3.378 nM T64567 CSW7I0 70681986 Ki = 3.633 nM T64567 CP65RU 70681987 Ki = 2.901 nM T64567 CFT68C 70681988 Ki = 3.679 nM T64567 C2Y5KV 70682044 Ki = 210 nM T64567 CR0D9S 70684100 Ki = 3.934 nM T64567 CRZ8S1 70684101 Ki = 3.592 nM T64567 COS95H 70684102 Ki = 3.633 nM T64567 CT5PH1 70684103 Ki = 3.156 nM T64567 C9P4BK 70685635 Ki = 757 nM T64567 C5XTY9 70686245 Ki = 3.554 nM T64567 C4SCY0 70688360 Ki = 3.311 nM T64567 CPD1N7 70688361 Ki = 2.863 nM T64567 C4L2OE 70688362 Ki = 2.758 nM T64567 CZO9C5 70688363 Ki = 3.429 nM T64567 CAD39I 70688364 Ki = 3.457 nM T64567 C7N4RT 70690386 Ki = 3.73 nM T64567 CQD8R9 70690387 Ki = 3.554 nM T64567 C1T4JL 70690936 Ki = 720 nM T64567 CUY3O8 70690937 Ki = 9240 nM T64567 CXF59L 70692549 Ki = 3.633 nM T64567 CV76WB 70692550 Ki = 3.73 nM T64567 C89LCZ 70692551 Ki = 3.403 nM T64567 C1K8VS 70692552 Ki = 3.679 nM T64567 CO5JP7 70692553 Ki = 3.633 nM T64567 CK5Y7G 70692554 Ki = 3.186 nM T64567 CGD06J 70692555 Ki = 3.378 nM T64567 C5QOK4 70692556 Ki = 3.633 nM T64567 C4BDK3 70694601 Ki = 3.788 nM T64567 CW8YA7 70694602 Ki = 2.573 nM T64567 CCYE61 70694603 Ki = 3.077 nM T64567 CEF1J8 70694604 Ki = 2.807 nM T64567 C4C0HK 70694605 Ki = 3.788 nM T64567 CBDQ72 70694606 Ki = 3.679 nM T64567 C95YWO 70695124 Ki = 6120 nM T64567 CSH7P1 70696148 Ki = 25.9 nM T64567 CWSA94 70696638 Ki = 3.52 nM T64567 CREC06 70696639 Ki = 3.679 nM T64567 CJ4M9S 70696640 Ki = 3.253 nM T64567 CHFY23 70696641 Ki = 3.73 nM T64567 C3Z7ER 70696642 Ki = 2.741 nM T64567 C6E4UW 70696643 Ki = 3.52 nM T64567 C0SP9E 70696644 Ki = 3.457 nM T64567 CAFH02 70696645 Ki = 3.855 nM T64567 CWQM13 70696646 Ki = 3.788 nM T64567 C04HIK 70698419 Ki = 6830 nM T64567 C8FB0P 71273627 Ki = 2.642 nM T64567 CJH6Y7 71273628 Ki = 3.355 nM T64567 CXG0H9 71273629 Ki = 3.031 nM T64567 CUT6R1 71273630 Ki = 3.633 nM T64567 CH49BT 71273631 Ki = 3.355 nM T64567 CK2U8R 71273632 Ki = 3.429 nM T64567 C2F9PC 71273633 Ki = 3.311 nM T64567 CV8FW3 71273635 Ki = 2.472 nM T64567 CQJ61A 71273738 Ki = 2.551 nM T64567 CSMV41 71273739 Ki = 3.311 nM T64567 CYW59B 71273740 Ki = 3 nM T64567 CU0KV6 71273743 Ki = 3.633 nM T64567 CC21VR 71273744 Ki = 3.592 nM T64567 C80KUG 71273750 Ki = 3.429 nM T64567 CJHN78 71415156 Ki = 220 nM T64567 CRN2O1 71449118 Ki = 28 nM T64567 C16PMU 71449958 IC50 = 9650 nM T64567 CXJ16H 71450117 Ki = 2340 nM T64567 CR79UB 71450332 Ki = 86.4 nM T64567 CT8E7N 71451561 Ki = 57 nM T64567 CHI2Z6 71452138 Ki = 11.8 nM T64567 CNI0R5 71452603 Ki = 77.8 nM T64567 C4E6PS 71453593 IC50 = 9900 nM T64567 CP27AT 71453970 Ki = 31 nM T64567 CW49YT 71453971 Ki = 29.7 nM T64567 C52WNJ 71454366 Ki = 85.1 nM T64567 CT90CD 71454373 Ki = 21.2 nM T64567 CB8JA3 71455488 Ki = 2570 nM T64567 C02UHX 71455489 Ki = 2182 nM T64567 CZ0S7D 71455712 Ki = 38.6 nM T64567 CUX07I 71455715 Ki = 60.6 nM T64567 C9COK3 71456113 Ki = 54.7 nM T64567 CICJ97 71457274 Ki = 1845 nM T64567 CL2BN6 71457492 Ki = 56.1 nM T64567 C4L0BG 71457918 Ki = 60.1 nM T64567 CWHN25 71459359 Ki = 65.2 nM T64567 CE31LC 71459360 Ki = 70.3 nM T64567 C70MBK 71459826 Ki = 67.2 nM T64567 C95MKT 71459827 Ki = 50.1 nM T64567 C5WYI8 71459828 Ki = 72.5 nM T64567 CD93TU 71461134 Ki = 66.3 nM T64567 C3WKX5 71461135 Ki = 71.2 nM T64567 C3YSR8 71461136 Ki = 93.4 nM T64567 CS1WI7 71461542 Ki = 23.1 nM T64567 C7VQ1R 71461543 Ki = 16.5 nM T64567 C4X1BZ 71462495 IC50 = 9100 nM T64567 CUM2H8 71462868 Ki = 76.2 nM T64567 CU4N0L 71462869 Ki = 17.3 nM T64567 C9KZA2 71462872 Ki = 33.4 nM T64567 CI6V9W 71489159 Ki = 470 nM T64567 CDQ8Z3 71498310 IC50 > 104 nM T64567 CIE7T0 71498311 IC50 = 4.42 nM T64567 CN6K9Q 71498738 IC50 = 42.23 nM T64567 CX6JP1 71498761 IC50 = 18.98 nM T64567 C98SLI 71498762 IC50 = 25.75 nM T64567 CJ2TX7 71498763 IC50 = 25.5 nM T64567 C0QX8S 71498764 IC50 = 54.35 nM T64567 CMHG14 71521493 Ki = 5900 nM T64567 CHN53G 71521494 Ki = 3300 nM T64567 CZJ5M6 71521495 Ki = 2900 nM T64567 CFBE53 71521496 Ki = 4500 nM T64567 CME27W 71521497 Ki = 9200 nM T64567 C24XWU 71521575 Ki = 5200 nM T64567 CJF68W 71521576 Ki = 8200 nM T64567 CHL8P3 71522144 Ki = 46 nM T64567 CEYG83 71522162 Ki = 3770 nM T64567 CZ78YT 71522163 Ki = 3260 nM T64567 C8NAF3 71545047 Ki = 29 nM T64567 C4H6PD 71545048 Ki = 950 nM T64567 CQ20AS 71545049 Ki = 86 nM T64567 CG2CL6 71545050 Ki = 60 nM T64567 C1MET8 71545051 Ki = 58 nM T64567 CILC35 71545052 Ki = 25 nM T64567 CGQ97W 71545216 Ki = 74 nM T64567 C71UMX 71545217 Ki = 18 nM T64567 C3KJ6D 71545218 Ki = 48 nM T64567 C0JNF3 71545219 Ki = 49 nM T64567 CC5EB7 71570660 Ki = 43.65 nM T64567 CA82YW 71570661 Ki = 11.37 nM T64567 CNL58G 71570662 Ki = 24.95 nM T64567 CDGY15 71578422 Ki = 66.9 nM T64567 CA5M6S 71578423 Ki = 32.2 nM T64567 CGOR42 71578424 Ki = 82.5 nM T64567 C45YXJ 71578425 Ki = 17.1 nM T64567 C1CKL6 71578426 Ki = 49.8 nM T64567 CR38IX 71578427 Ki = 86 nM T64567 CQ8Z5T 71578500 Ki = 7.8 nM T64567 CZ1R3F 71578570 Ki = 0.65 nM T64567 CV0G1A 71578571 Ki = 4.9 nM T64567 CX7T2V 71578640 Ki = 0.33 nM T64567 COT80J 71578641 Ki = 13 nM T64567 CGV68Z 71578723 Ki = 27 nM T64567 C7U0LV 71578724 Ki = 26 nM T64567 C8M0YB 71578725 Ki = 32 nM T64567 C4F0HB 71578726 Ki = 254 nM T64567 CZ29IK 71578808 Ki = 17 nM T64567 C8HMK5 71578809 Ki = 19 nM T64567 CMH2W4 71578810 Ki = 30 nM T64567 C7W9BS 71578811 Ki = 27 nM T64567 CU6N9T 71578812 Ki = 1857 nM T64567 CGEJ87 71578813 Ki = 23 nM T64567 C8CM0Q 71578898 Ki = 19 nM T64567 C19JFD 71578899 Ki = 29 nM T64567 C0MT2F 71578903 Ki = 157 nM T64567 CB9R7F 71578904 Ki = 21 nM T64567 CVTN91 71578980 Ki = 43.5 nM T64567 CBJ18U 71578981 Ki = 3462 nM T64567 CCKJ51 71578982 Ki = 83 nM T64567 C0TKR8 71579053 Ki = 90 nM T64567 CX4D6V 71579054 Ki = 2471 nM T64567 CJ0UP9 71579055 Ki = 47 nM T64567 CREN23 71579056 Ki = 2471 nM T64567 CP61GE 71579057 Ki = 2123 nM T64567 CXD68U 71579058 Ki = 73.2 nM T64567 C19OIY 71579130 Ki = 700 nM T64567 CV0LU6 71602117 Ki = 310 nM T64567 CCE15B 71602410 Ki = 29.3 nM T64567 CCB72P 71602411 Ki = 2.6 nM T64567 CHL16T 71602412 Ki = 5.9 nM T64567 C2UQV5 71602471 Ki = 3.1 nM T64567 C8K1YM 71602472 Ki = 2.4 nM T64567 CZL96Y 71602476 Ki = 3.1 nM T64567 CE70AQ 71602537 Ki = 8837 nM T64567 C3KPA8 71602538 Ki = 5.9 nM T64567 CO6FJ4 71602539 Ki = 2.9 nM T64567 CQ17LM 71602540 Ki = 4.6 nM T64567 C78LKP 71607884 IC50 = 3930 nM T64567 COVC80 71607885 IC50 > 3900 nM T64567 C1MOS8 71607912 IC50 > 690 nM T64567 CE0F4T 71607913 IC50 > 690 nM T64567 CO2LM4 71607914 IC50 > 690 nM T64567 CNBK57 71607915 IC50 > 690 nM T64567 CXPO21 71607916 IC50 = 690 nM T64567 CU24SZ 71607951 IC50 = 3.3 nM T64567 CJQW86 71607952 IC50 = 18.5 nM T64567 CR7BQ5 71607953 IC50 = 28.3 nM T64567 CPM89A 71607954 IC50 = 29 nM T64567 C1OPS4 71658869 Ki = 221 nM T64567 CN2FZ3 71659103 Ki > 50000 nM T64567 CC0EU9 71677604 Ki = 7.6 nM T64567 CS4VW3 71681364 Ki = 47.2 nM T64567 C5SY2L 71681517 Ki = 831 nM T64567 CT1D0W 71681519 Ki = 622 nM T64567 CW65GP 71681521 Ki = 765 nM T64567 CFS62D 71681523 Ki = 58 nM T64567 C96OCT 71681525 Ki = 4.3 nM T64567 C57BRD 71681527 Ki = 776 nM T64567 CU45ER 71681529 Ki = 779 nM T64567 C7NMJ2 71714066 Ki = 32600 nM T64567 C5DEF6 71714067 Ki = 15700 nM T64567 C50LSJ 71714068 Ki = 3570 nM T64567 C84WSV 71716939 Ki = 275 nM T64567 CBY8J3 71716994 Ki = 4400 nM T64567 CM4T1R 71717003 Ki = 3270 nM T64567 CN76CQ 71717054 Ki = 49 nM T64567 CI0SY3 71717570 Ki = 300 nM T64567 CYGT30 71717571 Ki = 324 nM T64567 CA3RM0 71717695 Ki = 900 nM T64567 CG4I1X 71718239 Ki = 710 nM T64567 C4N3VH 71718790 Ki = 2.656 nM T64567 C4B8KN 71718888 Ki = 66 nM T64567 C7U6NR 71719377 Ki = 375 nM T64567 CM24ND 71719433 Ki = 790 nM T64567 CT3D5S 71719441 Ki = 6700 nM T64567 CY3CV6 71719496 Ki = 48 nM T64567 CJG34A 71720036 Ki = 9750 nM T64567 CIU4L2 71720670 Ki = 830 nM T64567 CN0L8Q 71720672 Ki = 136 nM T64567 CY54DH 71728127 Ki > 10000 nM T64567 C9JAE7 71728128 Ki > 10000 nM T64567 C6HOP3 71728129 Ki > 10000 nM T64567 CRY5D8 71728130 Ki > 10000 nM T64567 CM91JE 71728236 Ki > 10000 nM T64567 C30ZEI 71728237 Ki > 10000 nM T64567 C4JB8W 71728238 Ki > 10000 nM T64567 C5RS9P 71728239 Ki > 10000 nM T64567 CRYC54 71728240 Ki > 10000 nM T64567 C5TKY7 71764398 Ki = 0.44 nM T64567 CMD91U 71764399 Ki = 7.2 nM T64567 CXO1T9 71764400 Ki = 7.8 nM T64567 CVEI80 71764401 Ki = 1.6 nM T64567 CVQ1H3 71764402 Ki = 1.8 nM T64567 CRZ64M 71764403 Ki = 10.1 nM T64567 CC0X1H 71764607 Ki = 6.3 nM T64567 CK7NI0 71764608 Ki = 0.74 nM T64567 C90YMG 71764609 Ki = 0.41 nM T64567 CK35HL 71764610 Ki = 5 nM T64567 C4SV1I 71764611 Ki = 1.2 nM T64567 C8NG9B 71764612 Ki = 0.52 nM T64567 CA2M1B 71764613 Ki = 0.62 nM T64567 CR7J6M 71764825 Ki = 1 nM T64567 CG09CJ 71764826 Ki = 0.57 nM T64567 CK2N0Z 71764827 Ki = 2.1 nM T64567 C08RAW 71765040 Ki = 1.3 nM T64567 CGI1J3 71765041 Ki = 0.61 nM T64567 CPT1X2 71765042 Ki = 0.31 nM T64567 C0ROQ1 71770179 Ki = 284 nM T64567 CGA62Y 71770789 Ki = 7.2 nM T64567 C8GP3J 71770790 Ki = 560 nM T64567 C04WFV 71770791 Ki = 43.6 nM T64567 CN4QC0 71770911 Ki = 713 nM T64567 C6XSA1 71770912 Ki = 6.4 nM T64567 C5YU4I 71770913 Ki = 101 nM T64567 C4G3HO 71770914 Ki = 89.1 nM T64567 CSU93P 71770915 Ki = 10.9 nM T64567 C9NAK1 71770916 Ki = 29.4 nM T64567 C42KOE 71770917 Ki = 63.5 nM T64567 CE8IC7 71770918 Ki = 395 nM T64567 CQJI19 71771031 Ki = 81.9 nM T64567 C2ZOB7 71771032 Ki = 5.4 nM T64567 C93LEJ 71771033 Ki = 140 nM T64567 C5UZM3 71771034 Ki = 811 nM T64567 CX9N5F 71818212 Ki = 35.3 nM T64567 C5IU0Y 72163201 Ki = 9.1 nM T64567 C0Q5XL 72163343 Ki = 12.3 nM T64567 C63MIX 72163344 Ki = 15.9 nM T64567 CL3WV2 72163345 Ki = 24 nM T64567 C4T9DA 72163346 Ki = 234 nM T64567 CTK07O 72163347 Ki = 9.4 nM T64567 CE32BF 72163348 Ki = 8.5 nM T64567 CA1X6Z 72163476 Ki = 8.8 nM T64567 C0FM1E 72202020 Ki = 376 nM T64567 CT41SJ 72202021 Ki = 41 nM T64567 C12SEI 72203721 IC50 = 91 nM T64567 CR37YX 72203722 IC50 = 138 nM T64567 C4VS2P 72203723 IC50 = 188 nM T64567 CSFR32 72203724 IC50 = 124 nM T64567 CDC0A4 72203725 IC50 = 141 nM T64567 CHUS18 72203726 IC50 = 84 nM T64567 C75RNW 72203906 IC50 = 34 nM T64567 C9AJ0V 72203907 IC50 = 51 nM T64567 C70JFO 72203908 IC50 = 74 nM T64567 CYKE59 72203909 IC50 = 90 nM T64567 CC1SO2 72203951 Ki = 44.4 nM T64567 CE9Q6G 72203952 Ki = 53.1 nM T64567 C5YJK2 72203953 Ki = 37.4 nM T64567 CCGB04 72204081 IC50 = 24 nM T64567 CR8I0V 72204082 IC50 = 85 nM T64567 C6X9ZV 72204083 IC50 = 87 nM T64567 CI5BS4 72204084 IC50 = 50 nM T64567 C72IXW 72204085 IC50 = 67 nM T64567 C3L1TY 72204086 IC50 = 52 nM T64567 CM2F7D 72204122 Ki = 2.2 nM T64567 C8XDF6 72204123 Ki = 4.7 nM T64567 CO51BD 72204124 Ki = 9.2 nM T64567 CWJE09 72204125 Ki = 19.4 nM T64567 C8XVK1 72204126 Ki = 13.5 nM T64567 CL54HN 72204268 IC50 = 43 nM T64567 CQ7U9H 72204269 IC50 = 48 nM T64567 C7WDI2 72204321 Ki = 20.93 nM T64567 CX4G0R 72204928 IC50 > 10000 nM T64567 CG9C6U 72204929 IC50 > 10000 nM T64567 C5A6XZ 72204930 IC50 > 10000 nM T64567 C0XZK4 72204931 IC50 > 10000 nM T64567 C6RY4X 72204933 IC50 > 10000 nM T64567 C4N5AB 72204934 IC50 > 10000 nM T64567 C3H2FZ 72205111 IC50 = 8234 nM T64567 CQ0VX7 72205112 IC50 > 10000 nM T64567 CQ7TI1 72205113 IC50 = 8210 nM T64567 CPAW52 72205114 IC50 = 8232 nM T64567 C2LD3J 72205115 IC50 = 8167 nM T64567 C4E2VS 72543811 Ki = 15.4 nM T64567 C3UJ8A 72695827 Ki = 9.2 nM T64567 CX82JD 72696463 Ki = 21.8 nM T64567 COCV73 72696591 Ki = 22.3 nM T64567 C5KHD7 72696592 Ki = 208 nM T64567 C4FBA6 72696593 Ki = 228 nM T64567 CO1JM5 72696594 Ki = 199 nM T64567 CUF61Q 72696595 Ki = 214 nM T64567 C1SU0Q 72712917 Ki = 8.3 nM T64567 COD5F4 72712918 Ki = 41 nM T64567 CJW7K4 72712919 Ki > 20000 nM T64567 CT2J8A 72712920 Ki > 20000 nM T64567 CRGC51 72713105 Ki = 21 nM T64567 C61VGR 72713106 Ki = 7.3 nM T64567 C96WHB 72713107 Ki = 8.3 nM T64567 CHPN94 72713108 Ki = 7.8 nM T64567 CJB8R7 72792832 Ki = 475 nM T64567 C5F7DT 72792833 Ki = 633 nM T64567 CAC7J8 72792834 Ki = 951 nM T64567 CFS02B 72792835 Ki = 426 nM T64567 CF5LW1 72792901 Ki = 78.1 nM T64567 C42IFJ 72792902 Ki = 480 nM T64567 CRMF25 72792903 Ki = 874 nM T64567 C2G5SR 72792904 Ki = 583 nM T64567 C6DR9O 72792905 Ki = 402 nM T64567 CGF5O1 72792967 Ki = 724 nM T64567 CWH3N9 72792968 Ki = 5.1 nM T64567 C5DSF8 72792969 Ki = 51.8 nM T64567 C2K6UZ 72792970 Ki = 335 nM T64567 CGI8K5 72793036 Ki = 374 nM T64567 C8WO6Z 72793037 Ki = 590 nM T64567 C6OZ0L 72793038 Ki = 943 nM T64567 CDTQ64 72793039 Ki = 126 nM T64567 CY16FM 72793040 Ki = 69.2 nM T64567 CXQN80 72793101 Ki = 800 nM T64567 CJ19BH 72793102 Ki = 254 nM T64567 CO1JT3 73054728 Ki = 9.8 nM T64567 C4MIP9 73345840 Ki = 760 nM T64567 C4Z7PY 73346473 Ki = 45.1 nM T64567 C48AKL 73346474 Ki = 341 nM T64567 CY2AH8 73346475 Ki = 78.3 nM T64567 C8QJU7 73346691 Ki = 6.8 nM T64567 C0PA8K 73346692 Ki = 6.3 nM T64567 CT6C3G 73346693 Ki = 7.3 nM T64567 CVN4A3 73346695 Ki = 14 nM T64567 CM9K3D 73346697 Ki = 12 nM T64567 C3Y4VZ 73347324 Ki = 3.2 nM T64567 C1WQ0C 73347968 Ki = 89.4 nM T64567 CEHI16 73348197 Ki = 8.2 nM T64567 C18GUI 73348198 Ki > 1000 nM T64567 C3CJ0F 73349055 Ki > 10000 nM T64567 C75IEZ 73349056 Ki > 10000 nM T64567 CK7MD1 73349516 Ki = 19.5 nM T64567 CJRE74 73349517 Ki = 31.7 nM T64567 CK98JL 73349518 Ki = 652 nM T64567 C6S7RY 73349758 Ki = 10 nM T64567 C2JP5U 73349759 Ki = 29.75 nM T64567 CBL42E 73350409 Ki = 3.3 nM T64567 CP3E7Q 73350410 Ki = 2.7 nM T64567 C38QDY 73351066 Ki = 24.8 nM T64567 COM17Y 73351067 Ki = 148 nM T64567 CN96PE 73351280 Ki = 7.5 nM T64567 CX1J7D 73352124 Ki > 10000 nM T64567 CXJL10 73352125 Ki > 10000 nM T64567 CBN25I 73352538 Ki = 65.4 nM T64567 CRDB68 73352539 Ki = 135 nM T64567 C4SNT8 73352540 Ki = 548 nM T64567 C3M2UH 73354029 Ki = 136 nM T64567 CB7Z2K 73355560 Ki = 23.1 nM T64567 CR81ON 73355561 Ki = 48.6 nM T64567 C60FZE 73355562 Ki = 239 nM T64567 CAK9J2 73355834 Ki = 15 nM T64567 CC2P6U 73356651 Ki > 10000 nM T64567 CC9AE6 73356652 Ki > 10000 nM T64567 C3SB2W 73357104 Ki = 124 nM T64567 C79KVE 73357105 Ki = 113 nM T64567 COP7H8 73357339 Ki = 8.1 nM T64567 CA3YT9 73894059 Ki = 2.4 nM T64567 C53JCV 74766009 Ki = 9 nM T64567 C53PBO 74766010 Ki = 24.3 nM T64567 CLPY57 74766011 Ki = 9.5 nM T64567 C7EF5V 76310135 Ki = 33 nM T64567 CLX6H0 76310136 Ki = 16 nM T64567 C9K6XP 76310137 Ki = 18 nM T64567 CX0Y6K 76310141 Ki = 316 nM T64567 C54AJY 76310148 Ki = 4.7 nM T64567 CCD80R 76310490 Ki = 8.7 nM T64567 CUB9V2 76310833 Ki = 115 nM T64567 C4S3QC 76310834 Ki = 114 nM T64567 CY7AV1 76310835 Ki = 22 nM T64567 CTJ50C 76310908 Ki > 50000 nM T64567 CEWJ18 76310909 Ki = 270 nM T64567 CR9G4Q 76311013 Ki = 8.4 nM T64567 CE7O5U 76311014 Ki = 12.4 nM T64567 CV19YL 76311015 Ki = 10 nM T64567 CO0PZ4 76311101 Ki = 7.8 nM T64567 CGT0J3 76311102 Ki = 9.1 nM T64567 CG2JI0 76313836 Ki = 15 nM T64567 CD1A5Y 76313837 Ki = 10.3 nM T64567 CU48XE 76313838 Ki = 30 nM T64567 C04EFJ 76313840 Ki = 78 nM T64567 CZ60NF 76313841 Ki = 355 nM T64567 C5S3XY 76313842 Ki = 416 nM T64567 CK2LR8 76313848 Ki = 8.1 nM T64567 CI3WQ5 76313849 Ki = 13.5 nM T64567 C0KVD7 76314143 Ki = 8.5 nM T64567 CE1H8W 76314144 Ki = 8.8 nM T64567 C5EM0L 76314145 Ki = 6.5 nM T64567 C0T8HW 76314452 Ki = 356 nM T64567 CZ0JC7 76314453 Ki = 16 nM T64567 CC1Z6A 76314549 Ki > 50000 nM T64567 CA1F9S 76314550 Ki > 50000 nM T64567 CZBG52 76314647 Ki = 2.1 nM T64567 C4F7WP 76314648 Ki = 22.8 nM T64567 C95DKS 76314709 Ki = 7.9 nM T64567 C37XBL 76314710 Ki = 136 nM T64567 C2H7ZA 76314711 Ki = 8.3 nM T64567 C34MRW 76317361 Ki = 59 nM T64567 CXZU92 76317371 Ki = 9.4 nM T64567 CB1VD3 76317966 Ki = 19.3 nM T64567 C6GOE1 76318042 Ki = 2.8 nM T64567 CGQ67N 76318218 Ki = 5.5 nM T64567 CLC1H8 76318279 Ki = 60.6 nM T64567 CT7G2Z 76318280 Ki = 10.5 nM T64567 CCO80M 76318281 Ki = 9.5 nM T64567 CY5O9B 76318282 Ki = 9.6 nM T64567 CM5IV7 76318283 Ki = 7.2 nM T64567 C4DMY8 76318284 Ki = 7.4 nM T64567 CG8QV5 76318285 Ki = 9.2 nM T64567 CDGH94 76321081 Ki = 17 nM T64567 CQ5B4S 76321082 Ki = 28 nM T64567 C9U3LR 76321089 Ki = 259 nM T64567 CZ2RY8 76321096 Ki = 26 nM T64567 C82NGW 76321408 Ki = 7820 nM T64567 CWM9C3 76321409 Ki = 10000 nM T64567 C78KRT 76321425 Ki = 9.1 nM T64567 CJ20ZB 76321688 Ki = 18.3 nM T64567 CVT3O8 76321689 Ki = 21.4 nM T64567 CH36SX 76321755 Ki = 76 nM T64567 C8SZN7 76321756 Ki = 104 nM T64567 CP24WC 76321814 Ki = 310 nM T64567 CNP1B7 76321907 Ki = 2 nM T64567 C4YP7A 76321908 Ki = 6.9 nM T64567 CZ98LC 76324732 Ki = 9.5 nM T64567 CW87DO 76324733 Ki = 46 nM T64567 C5JXE8 76324738 Ki = 89 nM T64567 CUG2O8 76324739 Ki = 310 nM T64567 CLN0I8 76325020 Ki = 39.3 nM T64567 C35EUT 76325021 Ki = 6.9 nM T64567 CZQ93S 76325300 Ki = 10.2 nM T64567 CP3X6L 76325374 Ki = 9 nM T64567 CO79TZ 76325375 Ki = 21 nM T64567 CE1DM0 76325376 Ki = 13 nM T64567 CE3P4W 76325377 Ki = 41 nM T64567 C7ZJ9M 76325378 Ki = 5.7 nM T64567 CN6CY7 76325452 Ki > 50000 nM T64567 CUC3M2 76325547 Ki = 9.4 nM T64567 C1BC4A 76325548 Ki = 2.8 nM T64567 CQUE95 76325602 Ki = 9 nM T64567 CDO73V 76325603 Ki = 102 nM T64567 C0UK2H 76328279 Ki = 21 nM T64567 CCNB68 76328280 Ki = 138 nM T64567 C8AS9R 76328281 Ki = 18 nM T64567 C0CFZ1 76328574 Ki = 873 nM T64567 CYM2G9 76328575 Ki = 8352 nM T64567 CZ5X4W 76328576 Ki = 1636 nM T64567 CP3CN4 76328593 Ki = 65.9 nM T64567 CPJM79 76328853 Ki = 5.9 nM T64567 C6F4LU 76328915 Ki = 25 nM T64567 C5VW9J 76328916 Ki = 431 nM T64567 CEZ6A8 76328917 Ki = 89 nM T64567 CYD50A 76329098 Ki = 7.1 nM T64567 CB23PR 76329099 Ki = 16.3 nM T64567 C3QI6J 76329100 Ki = 5.8 nM T64567 CTF2G1 76329169 Ki = 93.1 nM T64567 CAE23D 76329170 Ki = 8.3 nM T64567 CKH0X7 76331969 Ki = 27 nM T64567 CO82ZX 76331970 Ki = 26 nM T64567 C5U7JI 76331976 Ki = 197 nM T64567 CYC39A 76331984 Ki = 14 nM T64567 CK73VH 76331985 Ki = 139 nM T64567 C68DOK 76332270 Ki = 68.6 nM T64567 CJN0W8 76332271 Ki = 27.1 nM T64567 C3ZGF1 76332272 Ki = 8.2 nM T64567 C6ENW5 76332521 Ki = 5.1 nM T64567 C4RPU5 76332522 Ki = 1.2 nM T64567 C14UQS 76332523 Ki = 21.2 nM T64567 CGLB34 76332602 Ki = 3.7 nM T64567 CP9SU7 76332603 Ki = 64 nM T64567 CG3U6D 76332757 Ki = 49.3 nM T64567 CSN84K 76332758 Ki = 2.3 nM T64567 COZ89H 76332830 Ki = 62.7 nM T64567 CFI5K7 76332831 Ki = 875 nM T64567 C5VN9Q 76332832 Ki = 67.1 nM T64567 C9W0HZ 76335546 Ki = 62 nM T64567 CZC97G 76335551 Ki = 268 nM T64567 CQKW51 76335889 Ki > 10000 nM T64567 CB53XC 76335911 Ki = 56.8 nM T64567 CP16NU 76336199 Ki = 6.5 nM T64567 C3P4ZB 76336200 Ki = 7.6 nM T64567 CLB17E 76336381 Ki = 17.1 nM T64567 CV1B6C 76336382 Ki = 5.2 nM T64567 CWFY73 76336452 Ki = 531 nM T64567 C2QC4D 76336453 Ki = 8.8 nM T64567 CH0OY6 78319159 Ki = 82 nM T64567 CC4F0A 78319160 Ki = 23.7 nM T64567 CO4IE9 78319161 Ki = 26.5 nM T64567 CY6LN4 78319162 Ki = 43.8 nM T64567 CU9I6V 82078731 Ki = 58.4 nM T64567 C5TB6O 82080973 Ki = 25.8 nM T64567 CX5WB9 82198349 Ki = 12.1 nM T64567 C6UZR9 82911195 Ki = 8.2 nM T64567 CVD64Q 83379931 Ki = 342 nM T64567 CR47YB 86047482 Ki = 58 nM T64567 C0P3OF 86047486 Ki = 62.9 nM T64567 CZ5HA6 86047495 Ki = 62.8 nM T64567 CTD2Y9 86276273 Ki = 34 nM T64567 CHY2O4 86276274 Ki = 37 nM T64567 CN7HU3 86288843 Ki > 50000 nM T64567 C5Y1WO 86288855 Ki > 50000 nM T64567 C76RBA 86298624 IC50 = 601 nM T64567 C93FKI 86298625 IC50 = 84 nM T64567 CVLU48 86298626 IC50 = 596 nM T64567 CR97VD 86692717 Ki = 7.7 nM T64567 C8PC3U 86692718 Ki = 6.9 nM T64567 C6HC8V 86692720 Ki = 55.7 nM T64567 CQ30FJ 86719933 Ki = 4 nM T64567 CH2X9D 88314331 Ki = 22.8 nM T64567 C3EYT4 88314336 Ki = 8 nM T64567 C1O5YX 90180909 Ki = 220 nM T64567 CIJ96H 90644155 IC50 = 234 nM T64567 CX7EW1 90644156 IC50 > 10000 nM T64567 CK5GZ4 90644157 IC50 > 10000 nM T64567 C7O1YN 90644158 IC50 = 90 nM T64567 CEN6C1 90644159 IC50 = 78 nM T64567 C8X9UZ 90644160 IC50 = 2670 nM T64567 C4QT6W 90644479 Ki = 15.8 nM T64567 C6XB9R 90644480 Ki = 21.7 nM T64567 C1KXA0 90644481 Ki = 18.9 nM T64567 C1ND2E 90644482 Ki = 12.5 nM T64567 CY4LZ9 90644483 Ki = 26 nM T64567 C2RQD9 90644484 Ki = 38 nM T64567 CZ0R6T 90644485 Ki = 76 nM T64567 C4G1BD 90644486 Ki = 31 nM T64567 CL7I9M 90644487 Ki = 27 nM T64567 CVMU79 90644488 Ki = 15.3 nM T64567 C6F5ZP 90644489 Ki = 3.9 nM T64567 CG85NB 90644490 Ki = 10.2 nM T64567 CCID31 90644491 Ki = 4.8 nM T64567 C3BPF8 90644492 Ki = 5.5 nM T64567 C7B5YR 90644493 Ki = 3.1 nM T64567 C9FCX5 90644494 Ki = 2.8 nM T64567 CQND72 90644495 Ki = 9.7 nM T64567 C4V9IZ 90644496 Ki = 6.6 nM T64567 C49VLZ 90644497 Ki = 13.8 nM T64567 CX2I9G 90644498 Ki = 15.1 nM T64567 C5MXJ4 90644499 Ki = 13.2 nM T64567 C2E7QM 90644500 Ki = 10.9 nM T64567 CR02MV 90644501 Ki = 4.7 nM T64567 C2SZ5P 90644502 Ki = 13.6 nM T64567 C86NMC 90644503 Ki = 7 nM T64567 C8W3PI 90644504 Ki = 7.1 nM T64567 CF12MK 90645415 Ki = 6.3 nM T64567 CJO6I7 90645416 Ki = 3.9 nM T64567 CU2K5R 90645417 Ki = 2.7 nM T64567 C58KIU 90645418 Ki = 2.4 nM T64567 CS0OX7 90645419 Ki = 2.7 nM T64567 CWD6P7 90645420 Ki = 3 nM T64567 CVY5P9 90645421 Ki = 3.1 nM T64567 CAL9C4 90645422 Ki = 2.6 nM T64567 C2EA9C 90645423 Ki = 2.8 nM T64567 C1FVA8 90645424 Ki = 11.7 nM T64567 CP27AX 90645425 Ki = 325 nM T64567 C8E4ZH 90645426 Ki = 49.6 nM T64567 C3SIA9 90645429 Ki = 2.7 nM T64567 C1E4FS 90645430 Ki = 3.1 nM T64567 COBQ09 90645431 Ki = 2.8 nM T64567 C7IU8K 90645432 Ki = 3.6 nM T64567 CW0L1D 90654798 Ki > 50000 nM T64567 CO2CU1 90654800 Ki = 824 nM T64567 CE54MK 90654802 Ki > 50000 nM T64567 CID9U2 90654804 Ki = 652 nM T64567 C27QHW 90654822 Ki = 466 nM T64567 C96OWE 90654823 Ki = 484 nM T64567 CZQ9E3 90654824 Ki = 89.7 nM T64567 CCPO43 90654825 Ki = 443 nM T64567 C4D2TM 90654826 Ki = 341 nM T64567 C48XBN 90654827 Ki = 47.8 nM T64567 CI8TG3 90654828 Ki = 95.7 nM T64567 C6GFZ0 90654829 Ki = 8.6 nM T64567 C3Z1GS 90654830 Ki = 49.5 nM T64567 C4JSW5 90655322 Ki = 25 nM T64567 C3QH0R 90655323 Ki = 13 nM T64567 CF0U7K 90655324 Ki = 30 nM T64567 CU31VY 90675933 Ki = 37.7 nM T64567 C2XWG7 90675934 Ki = 40.1 nM T64567 CH7R2B 90675935 Ki = 24.4 nM T64567 CORQ94 90675936 Ki = 28.1 nM T64567 CE39DC 90675937 Ki = 40.3 nM T64567 CSU5K2 90675938 Ki = 30.9 nM T64567 CE8S1J 90675939 Ki = 33.4 nM T64567 C1H9FB 90675940 Ki = 39.8 nM T64567 CPB36R 90675941 Ki = 38.1 nM T64567 C0CR6D 90681501 Ki = 1120 nM T64567 C28FLQ 91498333 Ki = 62.5 nM T64567 CE6LO5 91595667 Ki = 23.1 nM T64567 C3AYZ5 91811067 Ki = 91.2 nM T64567 CQF98O 91827503 Ki = 9.4 nM T64567 C3I6NV 91827505 Ki = 7.5 nM T64567 CW1P4E 91827506 Ki = 5.01 nM T64567 CE2OY1 91995964 Ki = 9.2 nM T64567 CX45AP 92044053 Ki = 8.1 nM T64567 CEH68Q 93972064 Ki = 8.9 nM T64567 C28QRZ 101564149 Ki > 100000 nM T64567 CE8GH2 101874826 Ki = 9.6 nM T64567 C4W9FG 101874827 Ki = 8.1 nM T64567 CY7G8A 101874828 Ki = 78.9 nM T64567 C1TM8I 101874829 Ki = 9.7 nM T64567 CVZ3L5 101874830 Ki = 68.4 nM T64567 C2H5FC 101876957 Ki = 154 nM T64567 CDGZ03 101879106 Ki = 41.6 nM T64567 CY6ER7 101879108 Ki = 138.7 nM T64567 CAC1W7 101913750 Ki = 417 nM T64567 CQX8K1 101913751 Ki = 615 nM T64567 CIP25Q 101913752 Ki = 93 nM T64567 CTY15S 101913753 Ki = 462 nM T64567 C49NEJ 101913754 Ki = 485 nM T64567 CW5Q7L 101913755 Ki = 3860 nM T64567 CE90SD 102138248 Ki = 251 nM T64567 CB1PK8 102151146 Ki = 29500 nM T64567 C0A6FY 102151151 Ki > 100000 nM T64567 CP1X9Y 102232756 Ki = 420 nM T64567 C1XV9H 102311866 Ki > 100000 nM T64567 CQBE51 102341119 Ki = 2 nM T64567 C2TX7A 102354117 Ki = 228 nM T64567 CK43QR 102405972 Ki = 753 nM T64567 C0CVO4 102480165 Ki > 100000 nM T64567 C6LUE5 109059506 Ki = 234 nM T64567 CUY64D 109061586 Ki = 23.6 nM T64567 CXN7Z8 110453853 Ki = 78.1 nM T64567 C6I0LD 112499923 Ki = 126 nM T64567 C8CFR6 112499924 Ki = 208 nM T64567 CUR4V8 114816322 Ki = 31.8 nM T64567 C3TZ9A 115950959 Ki = 2.3 nM T64567 CAO67C 118705769 Ki = 5.8 nM T64567 CW1D8A 118705770 Ki = 6.6 nM T64567 CTFB51 118705771 Ki = 4.8 nM T64567 C5NGT8 118705772 Ki = 3.9 nM T64567 C3G4ZN 118705773 Ki = 5.8 nM T64567 CBVD13 118705774 Ki = 6.3 nM T64567 C3KCZ6 118705775 Ki = 54.7 nM T64567 C5Z4QF 118705776 Ki = 54.5 nM T64567 CV4YN0 118705777 Ki = 71.1 nM T64567 C0IBQ8 118705778 Ki = 63.9 nM T64567 CH7LV5 118705779 Ki = 57.6 nM T64567 CU5SI9 118705780 Ki = 5037 nM T64567 C6IGP0 118705781 Ki = 63.6 nM T64567 C7ZE2H 118705782 Ki = 34.5 nM T64567 C47QFN 118705783 Ki = 110 nM T64567 CO1P3T 118705784 Ki = 47.9 nM T64567 CK8E5C 118705785 Ki = 49.8 nM T64567 CS9G2U 118705786 Ki = 32.3 nM T64567 C1XV9M 118705787 Ki = 10.8 nM T64567 C7GW3Q 118705788 Ki = 11.3 nM T64567 CUIS94 118706141 Ki = 7.3 nM T64567 CET19U 118706142 Ki = 6.4 nM T64567 C6FBG3 118706893 Ki = 260 nM T64567 C1CLV5 118706959 Ki = 216 nM T64567 CLA5I2 118706960 Ki = 265 nM T64567 C8GD4Y 118706961 Ki = 192 nM T64567 CB0E4N 118706962 Ki = 223 nM T64567 CPI7L3 118710135 Ki = 114.4 nM T64567 C05ZCN 118710136 Ki = 199 nM T64567 C45XHE 118710137 Ki = 252 nM T64567 C84YKV 118710138 Ki = 47 nM T64567 CFA76H 118710139 Ki > 20000 nM T64567 C0UWK2 118710140 Ki > 20000 nM T64567 CGJ59E 118710141 Ki = 47 nM T64567 C64BUR 118710142 Ki = 43 nM T64567 C1W2DB 118710143 Ki = 41 nM T64567 CZ4F3O 118710144 Ki = 41 nM T64567 CWR82N 118710145 Ki = 266.6 nM T64567 C7R5FO 118710146 Ki > 20000 nM T64567 CD8U1O 118710147 Ki = 249 nM T64567 C8YFH6 118710148 Ki = 284 nM T64567 CLPC68 118710149 Ki = 285 nM T64567 C8OH4V 118710150 Ki = 275 nM T64567 C6CAQ4 118710151 Ki > 20000 nM T64567 CS0G7T 118710152 Ki > 20000 nM T64567 C3NPF1 118710200 Ki = 309 nM T64567 C4YXF1 118710201 Ki = 5.7 nM T64567 C1B5QL 118710202 Ki = 15.3 nM T64567 CUJ42P 118710203 Ki = 16.8 nM T64567 CK23DF 118710598 Ki = 73.9 nM T64567 CS9MC2 118710599 Ki = 25.1 nM T64567 CW2D4O 118710600 Ki = 23.1 nM T64567 CTMF04 118710601 Ki = 30.4 nM T64567 CU2C9L 118710602 Ki = 24 nM T64567 CFCG50 118710603 Ki = 20.5 nM T64567 C2G5DI 118710604 Ki = 38.7 nM T64567 CY2S9V 118710605 Ki = 80.4 nM T64567 C5L6IK 118710606 Ki = 81.3 nM T64567 C6ZGB2 118711612 Ki = 3 nM T64567 CNS6L8 118711613 Ki = 5 nM T64567 CY0E8G 118711614 Ki = 6.9 nM T64567 CI71PW 118711615 Ki = 6.2 nM T64567 C1X7RI 118711616 Ki = 5.4 nM T64567 C7P6GM 118711617 Ki = 127 nM T64567 CYNA84 118711618 Ki = 10.5 nM T64567 CL38UN 118711619 Ki = 21.3 nM T64567 CGUV98 118711620 Ki = 24.8 nM T64567 CJ2UH6 118711621 Ki = 38.9 nM T64567 CH2RE7 118711622 Ki = 5.3 nM T64567 C1RWN4 118711623 Ki = 4.7 nM T64567 CR0I6S 118711624 Ki = 4.5 nM T64567 C8LQI3 118711625 Ki = 12.8 nM T64567 C5SEJ6 118711626 Ki = 13.6 nM T64567 C5TYE7 118711627 Ki = 10.4 nM T64567 C7ZOH6 118712658 Ki = 779 nM T64567 C19IXJ 118712659 Ki = 673 nM T64567 CD5MB4 118712660 Ki = 773 nM T64567 C0EPI8 118712661 Ki = 936 nM T64567 CZ18GD 118716360 Ki = 215 nM T64567 CX6F4B 118716361 Ki = 215 nM T64567 CO4K8Z 118716362 Ki = 2 nM T64567 CR8HX4 118716363 Ki = 2 nM T64567 CYH2P1 118716364 Ki = 2 nM T64567 C61BOY 118716365 Ki = 115 nM T64567 C8PJC3 118716366 Ki = 2 nM T64567 C9HP7J 118716367 Ki = 2 nM T64567 CTS52R 118716368 Ki = 11 nM T64567 CHI60Z 118716369 Ki = 2 nM T64567 CA1UY4 118716496 Ki = 62.4 nM T64567 CVR32C 118716497 Ki = 141 nM T64567 CT1RQ6 118716498 Ki = 90.3 nM T64567 CG10AC 118716499 Ki = 86.6 nM T64567 CV89MK 118716500 Ki = 91.1 nM T64567 C57YMW 118716501 Ki = 460 nM T64567 CQ73KL 118716502 Ki = 51.2 nM T64567 CXE59K 118716504 Ki = 849 nM T64567 CONM87 118716505 Ki = 171 nM T64567 CQ3I7N 118716509 Ki = 6 nM T64567 C72KER 118716510 Ki = 5.4 nM T64567 C0RJI1 118716511 Ki = 5.5 nM T64567 CFU0Z8 118716512 Ki = 5.3 nM T64567 CXU4D7 118716513 Ki = 6.5 nM T64567 C86KQZ 118716514 Ki = 488 nM T64567 C9HLA8 118716891 Ki = 90 nM T64567 CJ0YC9 118716892 Ki = 79 nM T64567 CJ8TZ3 118716893 Ki = 54 nM T64567 C0X1WQ 118716894 Ki = 44 nM T64567 CDG4L8 118716895 Ki = 47 nM T64567 CFD26B 118716950 Ki = 162 nM T64567 C20YBM 118716951 Ki = 197 nM T64567 C0V1ZT 118716952 Ki = 28 nM T64567 CH9BW0 118716953 Ki = 165 nM T64567 CXB89Y 118716954 Ki = 113 nM T64567 C8CKU2 118716955 Ki = 244 nM T64567 CF03IX 118716956 Ki = 193 nM T64567 CYN29C 118716960 Ki = 27.9 nM T64567 C4AC7H 118716961 Ki = 23.6 nM T64567 CJ9O3I 118716962 Ki = 18.5 nM T64567 C6RJ9W 118716964 Ki = 213 nM T64567 CMVW90 118716999 Ki = 9 nM T64567 CBKN39 118717000 Ki = 44 nM T64567 C6N8CF 118717001 Ki = 8 nM T64567 CL3P7I 118717002 Ki = 9 nM T64567 C2H0NP 118717003 Ki = 8 nM T64567 CXRD23 118719969 Ki = 74.6 nM T64567 C4Z6DI 118719970 Ki = 9.7 nM T64567 C2HJ4Y 118719971 Ki = 90.7 nM T64567 CD1OH8 118719972 Ki = 22.8 nM T64567 C0R8JN 118719973 Ki = 89.2 nM T64567 CMR0H2 118719974 Ki = 20.2 nM T64567 CI3QG5 118719975 Ki = 23.1 nM T64567 C06YTV 118719976 Ki = 87.8 nM T64567 C25BJT 118721385 Ki = 1747 nM T64567 CI4W0E 118721386 Ki = 699 nM T64567 CFRX59 118721387 Ki = 229 nM T64567 C5SYD7 118721388 Ki = 1022 nM T64567 CNT18B 118721389 Ki = 1692 nM T64567 CYC50E 118721390 Ki = 2109 nM T64567 CYL0W1 118721391 Ki = 752 nM T64567 C1HN6R 118721392 Ki = 109 nM T64567 C2WLI4 118721393 Ki = 842 nM T64567 CQVS30 118721394 Ki = 62.4 nM T64567 CL2Q8M 118721395 Ki = 2.8 nM T64567 CAG5L6 118721396 Ki = 60.4 nM T64567 CJ63BR 118721397 Ki = 81.6 nM T64567 C14ZNT 118721398 Ki = 186 nM T64567 C1J6IX 118721399 Ki = 111 nM T64567 CVJ92D 118721400 Ki = 739 nM T64567 C5F7PT 118721401 Ki = 224 nM T64567 C5AFR3 118721402 Ki = 854 nM T64567 C29EYL 118721403 Ki = 114 nM T64567 C8GYO9 118721404 Ki = 134 nM T64567 CSZ7Q0 118721405 Ki = 91.6 nM T64567 CY3ZW6 118721406 Ki = 224 nM T64567 C4T9IR 118721407 Ki = 152 nM T64567 CNPB81 118721408 Ki = 119 nM T64567 CP40JF 118722001 Ki = 42.4 nM T64567 CXTR97 118723294 Ki = 8.3 nM T64567 C42JBV 118723295 Ki = 5.8 nM T64567 CVDC56 118723296 Ki = 7.1 nM T64567 C2RG7F 118723303 Ki = 8.5 nM T64567 C0CMO4 118723304 Ki = 7.2 nM T64567 CC7RH0 118723305 Ki = 8.8 nM T64567 CU0R8X 118723306 Ki = 9.6 nM T64567 C67LPC 118723308 Ki = 7.9 nM T64567 C0D1SQ 118724328 Ki = 46 nM T64567 C89YTC 118724329 Ki = 456.6 nM T64567 CBT87C 118724330 Ki = 106.4 nM T64567 C49AWZ 118724331 Ki = 300.9 nM T64567 CP9X5K 118728047 Ki = 37.9 nM T64567 CUA3S7 118728048 Ki = 0.91 nM T64567 C2K3DO 118728049 Ki = 0.97 nM T64567 CZTN86 118728050 Ki = 2.6 nM T64567 C0CUV2 118728051 Ki = 93.5 nM T64567 CGU5O0 118728053 Ki = 71.8 nM T64567 CGQ69F 118728055 Ki = 82.4 nM T64567 C2JEW0 118728057 Ki = 72 nM T64567 CCBJ19 118728058 Ki = 67.1 nM T64567 CKJ8S9 118728060 Ki = 41.3 nM T64567 C0O3BI 118728062 Ki = 86.2 nM T64567 CH2E8F 118728064 Ki = 9.5 nM T64567 C4JM1O 118728066 Ki = 0.97 nM T64567 C67YPT 118728068 Ki = 55.1 nM T64567 CML9F8 118728070 Ki = 6.7 nM T64567 CA52IR 118728072 Ki = 79.9 nM T64567 CVE9H5 118728074 Ki = 0.91 nM T64567 CS9ZW3 118728500 Ki = 38.7 nM T64567 CI7MY8 118728501 Ki = 32.6 nM T64567 CZE9K8 118728502 Ki = 31.3 nM T64567 C8S9JV 118728503 Ki = 31.6 nM T64567 C40AIB 118729374 Ki = 59.9 nM T64567 CO3Z5E 118729375 Ki = 77.4 nM T64567 C6S0DR 118729376 Ki = 70.8 nM T64567 CVXO79 118729377 Ki = 95.3 nM T64567 C62BGK 118729378 Ki = 10.3 nM T64567 C4D9EP 118729379 Ki = 70.9 nM T64567 C2TOH7 118729380 Ki = 9.8 nM T64567 C5P9ND 118729381 Ki = 76.2 nM T64567 C2XLV4 118729382 Ki = 9.1 nM T64567 CVLK60 118729383 Ki = 29.7 nM T64567 C8U7SE 118729384 Ki = 9.8 nM T64567 CV7OS1 118729385 Ki = 9 nM T64567 C7Z2OR 118729386 Ki = 9.4 nM T64567 CHE1K4 118729473 Ki = 0.86 nM T64567 C9V8MA 118729474 Ki = 21.6 nM T64567 C8GJP5 118729475 Ki = 34.1 nM T64567 C4MEZ0 118729476 Ki = 10.3 nM T64567 CE3IV5 118729477 Ki = 9 nM T64567 C5DM9L 118731312 Ki = 6 nM T64567 C08EZC 118733945 Ki = 23.84 nM T64567 C3F1DU 118733947 Ki = 37.62 nM T64567 C4OL1A 118733948 Ki = 19.91 nM T64567 CP25HS 118733949 Ki = 32.09 nM T64567 CY3H4E 118736318 Ki = 231 nM T64567 C8HY4S 118736320 Ki = 123 nM T64567 C7F5JH 118736322 Ki = 230 nM T64567 C7MDJ3 118736324 Ki = 4.1 nM T64567 CQM67J 118736325 Ki = 3.7 nM T64567 CKY90W 118736326 Ki = 4.3 nM T64567 CY4B1U 118736327 Ki = 15.6 nM T64567 CRZ1T6 118736328 Ki = 4.1 nM T64567 CFDB97 118737265 Ki = 9.6 nM T64567 CVGF86 118737267 Ki = 17.2 nM T64567 C6B8WR 118737268 Ki = 5.6 nM T64567 CWEM68 118737269 Ki = 6.6 nM T64567 C6PXT8 118737270 Ki = 9 nM T64567 CWP7Q1 118737271 Ki = 9.7 nM T64567 CAB65M 118737272 Ki = 9.1 nM T64567 CHR0I7 118737273 Ki = 81.3 nM T64567 C72BLG 118737274 Ki = 29.5 nM T64567 C4TD0Q 118737275 Ki = 33 nM T64567 CZ1J0U 118737276 Ki = 10.5 nM T64567 CHN09Y 118737277 Ki = 7.7 nM T64567 CMR62B 118737278 Ki = 42.1 nM T64567 C1CV3E 118737279 Ki = 33.8 nM T64567 CUQ7H9 119082247 Ki = 2.7 nM T64567 CP8Y5U 119090745 Ki = 8.2 nM T64567 C4K6CG 119943184 Ki = 27 nM T64567 CHX4Y2 121382833 Ki > 50000 nM T64567 CNEJ87 121382878 Ki = 172 nM T64567 CBHM75 121382881 Ki = 4610 nM T64567 C13GKC 121382882 Ki = 2740 nM T64567 C8QTR4 121382883 Ki = 8970 nM T64567 C96ANJ 121382897 Ki > 50000 nM T64567 CUS64J 121382999 Ki = 271 nM T64567 C6C4WE 121383002 Ki = 176 nM T64567 CG48HD 122164592 Ki = 2910 nM T64567 CK92MV 122179845 Ki = 29.6 nM T64567 C10UQY 122179846 Ki = 28.7 nM T64567 CLV96C 122179847 Ki = 25.4 nM T64567 C2RT1Y 122179848 Ki = 24.5 nM T64567 C06ZSC 122179849 Ki = 13.8 nM T64567 C74RAE 122179850 Ki = 35.6 nM T64567 C6NM0Q 122179851 Ki = 27.7 nM T64567 CYP3B0 122179852 Ki = 26.6 nM T64567 CMP05I 122179853 Ki = 417 nM T64567 C2TGN6 122179854 Ki = 403 nM T64567 CAH3I1 122179855 Ki = 42.3 nM T64567 C8YJ9B 122180166 Ki = 151 nM T64567 CHON20 122180167 Ki = 2024 nM T64567 C9L2TG 122180168 Ki = 213 nM T64567 C9L3OY 122180169 Ki = 1256 nM T64567 CJ1X2F 122180170 Ki = 110 nM T64567 CVCX92 122180171 Ki = 2037 nM T64567 C6LEA3 122180172 Ki = 246 nM T64567 CV8Z4I 122182643 Ki = 172 nM T64567 CV96QP 122182644 Ki = 244 nM T64567 CA91HP 122182645 Ki = 67.3 nM T64567 C08EBQ 122182646 Ki = 135 nM T64567 CSJA24 122182647 Ki = 4.8 nM T64567 CDM51W 122182648 Ki = 276 nM T64567 C3E9FK 122182649 Ki = 295 nM T64567 CUF5N9 122182650 Ki = 2.8 nM T64567 C5BRH0 122182651 Ki = 2.7 nM T64567 C45DQE 122182654 Ki = 2.8 nM T64567 CDRF43 122182655 Ki = 3.9 nM T64567 CQ83BJ 122182656 Ki = 2.1 nM T64567 CH4Z8B 122182657 Ki = 2.6 nM T64567 CU71LK 122182658 Ki = 2.5 nM T64567 CY1NK4 122182659 Ki = 2.3 nM T64567 CP4I8D 122184891 Ki = 71.6 nM T64567 CZ2RM0 122184892 Ki = 70.7 nM T64567 CFQ4R3 122184893 Ki = 52.4 nM T64567 C69UQF 122184894 Ki = 44.7 nM T64567 CNF20A 122184895 Ki = 32.9 nM T64567 CJAL95 122184896 Ki = 44.4 nM T64567 C51LFX 122184933 Ki = 63.1 nM T64567 CTQP23 122184934 Ki = 67.1 nM T64567 CL49QM 122184935 Ki = 56.9 nM T64567 CVN28C 122184936 Ki = 6.9 nM T64567 CU4S6Y 122184937 Ki = 30.8 nM T64567 C4VWG9 122184938 Ki = 67.2 nM T64567 C7H8ZI 122184984 Ki = 10.5 nM T64567 CX76HF 122184985 Ki = 11.1 nM T64567 C1KOF6 122184986 Ki = 61.5 nM T64567 C01CWK 122184987 Ki = 10.4 nM T64567 CVTY87 122184988 Ki = 0.91 nM T64567 CM5A7F 122184989 Ki = 32.3 nM T64567 CYM65N 122184990 Ki = 34.1 nM T64567 CQ9YU1 122184991 Ki = 114.1 nM T64567 C83GXC 122184992 Ki = 113.6 nM T64567 CTV40W 122184993 Ki = 24.3 nM T64567 CWM21G 122184994 Ki = 6.7 nM T64567 C19LDQ 122184995 Ki = 120.7 nM T64567 C7UE2C 122184996 Ki = 36.9 nM T64567 CWBN52 122184997 Ki = 80.5 nM T64567 C1CI4W 122184998 Ki = 549.2 nM T64567 CWJ94V 122185033 Ki = 2 nM T64567 C9PG8Z 122185234 Ki = 277 nM T64567 C93KBM 122185235 Ki = 353 nM T64567 CX6Z5Y 122185236 Ki = 274 nM T64567 CFPV38 122185237 Ki = 193 nM T64567 CVZ70D 122185238 Ki = 342 nM T64567 C14OHP 122185239 Ki = 29.5 nM T64567 CB63WU 122185240 Ki = 85.5 nM T64567 CE3Q1J 122185241 Ki = 29.4 nM T64567 CNG63S 122185242 Ki = 32.5 nM T64567 CY7H0T 122185243 Ki = 22.7 nM T64567 C2ME1I 122185244 Ki = 16.5 nM T64567 C0EPT7 122185245 Ki = 150 nM T64567 CI1AL4 122185246 Ki = 354 nM T64567 CM43CE 122185684 Ki = 26 nM T64567 CSQ43L 122185685 Ki = 210 nM T64567 CCA9I1 122185686 Ki = 25 nM T64567 CLIR24 122185687 Ki = 27 nM T64567 C5NWU9 122185688 Ki = 32 nM T64567 CY70TU 122185689 Ki = 31 nM T64567 CD94UC 122185690 Ki = 32 nM T64567 C8TIP4 122185692 Ki = 26 nM T64567 CE7W6O 122185694 Ki = 202 nM T64567 CV2G7S 122185695 Ki = 61 nM T64567 C1M5JR 122185696 Ki = 1.9 nM T64567 CMB32C 122185697 Ki = 15 nM T64567 C1FR9Q 122185698 Ki = 150 nM T64567 CY2D9L 122185699 Ki = 25 nM T64567 C2NUJ9 122185700 Ki = 23 nM T64567 CHBC74 122185771 Ki = 2.6 nM T64567 CZM98F 122185772 Ki = 21 nM T64567 CP8Y5E 122185773 Ki = 23 nM T64567 CK2Q7M 122185774 Ki = 27 nM T64567 CF4L0N 122185776 Ki = 20 nM T64567 C7T4BF 122185778 Ki = 28 nM T64567 C4TZ6G 122185779 Ki = 20 nM T64567 CUI73A 122187162 Ki = 3.2 nM T64567 C1Q7AX 122187163 Ki = 6.5 nM T64567 CO6P7A 122187164 Ki = 1.7 nM T64567 C9LN8Q 122187165 Ki = 1.6 nM T64567 COK6D7 122187166 Ki = 274 nM T64567 C7NV8G 122187167 Ki = 318 nM T64567 C6XKH1 122187168 Ki = 285 nM T64567 C5KMW2 122187169 Ki = 276 nM T64567 CSA78D 122187170 Ki = 438 nM T64567 C5V7SZ 122187171 Ki = 3.1 nM T64567 C6FMG1 122187172 Ki = 42.5 nM T64567 CVG1U0 122187173 Ki = 3.7 nM T64567 CR8NT0 122187174 Ki = 4.1 nM T64567 CWSM36 122187175 Ki = 4.5 nM T64567 CT59AR 122187176 Ki = 10.5 nM T64567 C93ESN 122187177 Ki = 122 nM T64567 CL0JF6 122187178 Ki = 156 nM T64567 CQ81UP 122187179 Ki = 18.7 nM T64567 CIE0W8 122187180 Ki = 36.4 nM T64567 CNSU27 122187181 Ki = 26.3 nM T64567 C7LDH1 122187182 Ki = 13.1 nM T64567 CG9T3N 122187183 Ki = 25.9 nM T64567 CBE9U8 122187184 Ki = 15.2 nM T64567 C13USE 122187185 Ki = 28 nM T64567 CE36PK 122187423 Ki = 436 nM T64567 CDS2I6 122187424 Ki = 9.9 nM T64567 CMF63L 122187425 Ki = 320 nM T64567 C7Q9TP 122187426 Ki = 268 nM T64567 C04HSI 122187596 Ki = 57 nM T64567 CZ74KO 122187597 Ki = 77 nM T64567 C07OYV 122187598 Ki = 90 nM T64567 CO6AT2 122187599 Ki = 75 nM T64567 C7WJ4B 122187600 Ki = 75 nM T64567 CZ0Y1G 122187601 Ki = 86 nM T64567 CWF7Z0 122187602 Ki = 86 nM T64567 C07ZNW 122187603 Ki = 85 nM T64567 C7K6TV 122187604 Ki = 61 nM T64567 CX69YT 122187605 Ki = 91 nM T64567 C8XN0F 122187606 Ki = 74 nM T64567 CVT13C 122187607 Ki = 61 nM T64567 CB2DT8 122187638 Ki = 39.6 nM T64567 C0G4CQ 122187639 Ki = 129 nM T64567 CQSV13 122187640 Ki = 487 nM T64567 CH74EW 122187641 Ki = 280 nM T64567 CH3C8V 122187642 Ki = 202 nM T64567 CP01NQ 122187643 Ki = 134 nM T64567 CRM3S4 122188878 Ki = 84.3 nM T64567 C5UF1Q 122188879 Ki = 135 nM T64567 CQB9A8 122188880 Ki = 154 nM T64567 C1SFD4 122188881 Ki = 248 nM T64567 CIE7L0 122188882 Ki = 213 nM T64567 C6MPI4 122189078 Ki = 65 nM T64567 C9V7WT 122189088 Ki = 7.5 nM T64567 C1QZV7 122189098 Ki = 48.7 nM T64567 CN16RY 122189300 Ki = 17 nM T64567 CYN3T8 122189301 Ki = 6.1 nM T64567 CSW9D1 122189302 Ki = 27 nM T64567 C6USQ7 122189303 Ki = 28 nM T64567 CQ4X1G 122189304 Ki = 42 nM T64567 C5XT3S 122192640 Ki = 1020 nM T64567 C1LCB9 122192641 Ki = 1000 nM T64567 CP51XT 122192642 Ki = 920 nM T64567 C5GKT0 122192643 Ki = 580 nM T64567 C3RZM8 122192644 Ki = 100 nM T64567 CHLG86 122192645 Ki = 440 nM T64567 CTK4J8 122192646 Ki = 1120 nM T64567 CVNQ49 122192647 Ki = 90 nM T64567 CX3A0N 122192648 Ki = 280 nM T64567 CU3F1V 122192649 Ki = 110 nM T64567 CQ4NT8 122192650 Ki = 100 nM T64567 C2REU8 122192651 Ki = 800 nM T64567 CL5P4T 122192652 Ki = 250 nM T64567 C0KF5I 122192653 Ki = 90 nM T64567 CT64DB 122192654 Ki = 810 nM T64567 CX05RY 122192671 Ki = 24.9 nM T64567 CE9ZC4 122192672 Ki = 31.2 nM T64567 CUW2B9 122192673 Ki = 27.5 nM T64567 CKU76Q 122192674 Ki = 23.6 nM T64567 C49KGU 122192675 Ki = 24 nM T64567 CB0J2T 122192676 Ki = 23 nM T64567 CS63LF 122192677 Ki = 26.9 nM T64567 C4T3IO 122192678 Ki = 28.8 nM T64567 CTZ4L6 122192679 Ki = 14.3 nM T64567 C62VGD 122192680 Ki = 33.1 nM T64567 CYND20 122192681 Ki = 29.6 nM T64567 CLV5O9 122192682 Ki = 34.4 nM T64567 CH1N0C 122193189 Ki = 930 nM T64567 C19HVL 122193190 Ki = 970 nM T64567 C5TQJ1 122193251 Ki = 990 nM T64567 C8XCL0 122193252 Ki = 820 nM T64567 CH4IV8 122194771 Ki = 9.3 nM T64567 CQ7N0L 122194772 Ki = 71.4 nM T64567 CI5K2F 122194773 Ki = 823 nM T64567 CV51IU 122194774 Ki = 8.4 nM T64567 C7OFR6 122194775 Ki = 63.8 nM T64567 C81HNW 122194776 Ki = 8.9 nM T64567 C8J5QV 122194777 Ki = 519 nM T64567 CV1C9T 122194778 Ki = 42.3 nM T64567 CJC1W3 122194779 Ki = 710 nM T64567 CU1TV5 122194780 Ki = 76.7 nM T64567 C4C1BE 122194781 Ki = 450 nM T64567 CR9I5Q 122194782 Ki = 31.4 nM T64567 C8SVY4 122194783 Ki = 85.6 nM T64567 C7HT8B 122194784 Ki = 678 nM T64567 CW8P3R 122194785 Ki = 705 nM T64567 COAK34 122194786 Ki = 6 nM T64567 CPN73S 122199224 Ki = 39 nM T64567 CC1UO6 122226187 Ki = 9100 nM T64567 C7T0FH 122226188 Ki = 22900 nM T64567 C3EG2B 122226189 Ki = 37000 nM T64567 C18KAD 122367673 Ki > 50000 nM T64567 CPN5F4 122367675 Ki > 50000 nM T64567 C26IUP 122386532 Ki > 100000 nM T64567 CGE1Q6 122707121 Ki = 98.5 nM T64567 C1JBF7 122707123 Ki = 0.18 nM T64567 CGPI62 123372490 Ki = 28.1 nM T64567 CV4GW7 126961712 Ki = 32.7 nM T64567 C0FD4E 126961713 Ki = 39.2 nM T64567 CXY79J 127024883 Ki = 261 nM T64567 CK9C7T 127024884 Ki = 210 nM T64567 C50MSQ 127024885 Ki = 161 nM T64567 C4N6WJ 127024886 Ki = 2482 nM T64567 C5AES0 127024887 Ki = 26 nM T64567 CHU95V 127024991 Ki = 224 nM T64567 CP8O7D 127024992 Ki = 240 nM T64567 CRHW31 127024993 Ki = 0.17 nM T64567 C57BLH 127025130 Ki = 7.4 nM T64567 CRTB63 127025292 Ki = 159 nM T64567 CAO31Y 127025293 Ki = 216 nM T64567 CL0ZR4 127025295 Ki = 258 nM T64567 C9JNZ5 127025296 Ki = 0.24 nM T64567 C04USY 127025300 Ki = 35.6 nM T64567 CDB1Z9 127025301 Ki = 16.2 nM T64567 CYK6H1 127025302 Ki = 17.5 nM T64567 C7UF0B 127025480 Ki = 196 nM T64567 C6M4SW 127025591 Ki = 45 nM T64567 CUPA95 127025592 Ki = 3.7 nM T64567 CWP36V 127025593 Ki = 49.3 nM T64567 C95QVS 127026977 Ki = 40.8 nM T64567 C09PAM 127026978 Ki = 54.1 nM T64567 CS96JF 127026979 Ki = 335 nM T64567 CRB80M 127026980 Ki = 67.8 nM T64567 C0RBK5 127027010 Ki = 27 nM T64567 C0WY9H 127027097 Ki = 2.3 nM T64567 CP84DU 127027288 Ki = 92.7 nM T64567 CH30BV 127027289 Ki = 7 nM T64567 CM72RV 127027290 Ki = 22.5 nM T64567 CO3IJ7 127027291 Ki = 8.7 nM T64567 C4O2XT 127028951 Ki = 239 nM T64567 CFIW54 127029020 Ki = 124 nM T64567 C5RBS3 127029021 Ki = 156 nM T64567 CPA6G5 127029022 Ki = 0.37 nM T64567 C74ZGJ 127029023 Ki = 0.21 nM T64567 CN3PH9 127029250 Ki = 265 nM T64567 CTY1H9 127029498 Ki = 27.6 nM T64567 C1J0RU 127029568 Ki = 50.4 nM T64567 CS2K4U 127034999 Ki = 25.7 nM T64567 CFG39M 127035855 Ki = 30.5 nM T64567 C6MH2V 127035856 Ki = 29.3 nM T64567 CVO4B6 127035857 Ki = 26.5 nM T64567 CQC6P9 127035858 Ki = 117 nM T64567 C7YA3N 127035859 Ki = 96.7 nM T64567 CXZI89 127035860 Ki = 28.1 nM T64567 C5KLP8 127035861 Ki = 225 nM T64567 CTVN28 127036466 Ki = 8.1 nM T64567 CWPY69 127036947 Ki = 6.1 nM T64567 CL76JS 127037630 Ki = 191 nM T64567 CY1JU3 127037755 Ki = 52 nM T64567 CL3Q0T 127037870 Ki = 276 nM T64567 CK3VW1 127037881 Ki = 100 nM T64567 CTSR32 127038212 Ki = 5.1 nM T64567 CQTS23 127038553 Ki = 259 nM T64567 C6WCG5 127039856 Ki = 45.4 nM T64567 C4NQ5H 127039905 Ki = 163 nM T64567 C0P5HB 127040227 Ki = 43.9 nM T64567 CCD87Q 127040239 Ki = 275 nM T64567 C97DAS 127040240 Ki = 14.5 nM T64567 C9OZP8 127040553 Ki = 157 nM T64567 C4SH5D 127040554 Ki = 34.9 nM T64567 CCO9S8 127040555 Ki = 4.7 nM T64567 C12SMV 127041490 Ki = 0.22 nM T64567 CSJ3V0 127041732 Ki = 36.9 nM T64567 CG75VH 127041733 Ki = 24.3 nM T64567 C41YOV 127044252 Ki = 24.9 nM T64567 CMTC13 127044428 Ki = 554 nM T64567 C7KU0Z 127044429 Ki = 74.7 nM T64567 CJO3U8 127044444 Ki = 70.2 nM T64567 CAXM67 127044445 Ki = 641.5 nM T64567 CHP23N 127044446 Ki = 23.3 nM T64567 C0KQB1 127044932 Ki = 5.6 nM T64567 C62OLS 127045037 Ki = 6.7 nM T64567 C31FCL 127045083 Ki = 29.2 nM T64567 CT9KP2 127045237 Ki = 7.3 nM T64567 C17GLC 127045238 Ki = 8.8 nM T64567 C1U0VA 127045339 Ki = 49.3 nM T64567 CG10PI 127048878 Ki = 28.25 nM T64567 C3PHY8 127048879 Ki = 21.58 nM T64567 COLX43 127048880 Ki = 28.57 nM T64567 CBJ74P 127048881 Ki = 24.47 nM T64567 C1XE4W 127049197 Ki = 23.14 nM T64567 CCX35L 127049198 Ki = 25.04 nM T64567 CRE6O9 127049213 Ki = 25.96 nM T64567 CP40EB 127049242 Ki = 1.7 nM T64567 CLFB54 127049248 Ki = 2.5 nM T64567 CY5MI3 127049999 Ki = 420 nM T64567 C5CNP8 127050174 Ki = 19.73 nM T64567 CH07TV 127050456 Ki = 2.28 nM T64567 CP8U0D 127050457 Ki = 2.54 nM T64567 C65PAS 127050458 Ki = 26.53 nM T64567 CJP49X 127050777 Ki = 2.32 nM T64567 CER02F 127050778 Ki = 28.07 nM T64567 CG17IO 127050812 Ki = 4.8 nM T64567 C8X6CY 127050822 Ki = 3 nM T64567 C4IA5N 127051119 Ki = 2.9 nM T64567 CRDQ30 127051120 Ki = 9.6 nM T64567 CJ0EQ7 127051501 Ki > 50000 nM T64567 C5Y4DI 127051953 Ki = 24.1 nM T64567 CM21NF 127052276 Ki = 23.59 nM T64567 C90PLX 127052516 Ki = 8720 nM T64567 CFQ75A 127052517 Ki = 840 nM T64567 CEC30I 127052811 Ki = 2790 nM T64567 C5CW4K 127052812 Ki = 5990 nM T64567 C5V7QI 127052813 Ki = 2000 nM T64567 CI24ZM 127052900 Ki = 58.61 nM T64567 CEVZ36 127052901 Ki = 2.35 nM T64567 CX1Z2E 127052917 Ki = 21.64 nM T64567 CM8FI7 127052918 Ki = 20.4 nM T64567 CUOZ60 127052919 Ki = 20.08 nM T64567 CHN5K6 127567366 Ki = 3.9 nM T64567 C4JC3W 127573780 Ki = 0.7 nM T64567 C85FAK 129009671 Ki = 2.1 nM T64567 C7R6LY 129009672 Ki = 2.6 nM T64567 C2B6XM 129673327 Ki = 54.4 nM T64567 CJC35Q 129856021 Ki = 170.8 nM T64567 CCF61S 129883275 Ki = 58.7 nM T64567 CNB2M7 131839635 Ki = 5.3 nM T64567 C7Z4UB 132494202 Ki = 57.9 nM T64567 C20FGA 132495363 Ki = 10.9 nM T64567 C4GR3Y 132498655 Ki = 0.53 nM T64567 CKLY32 132502995 Ki = 4869 nM T64567 CJQP17 132541861 Ki = 2.7 nM T64567 CVM1A9 132547283 Ki = 275 nM T64567 C3H1NS 132547284 Ki = 2830 nM T64567 C1FWS2 132547285 Ki = 251 nM T64567 C7Z5LX 132547286 Ki = 143 nM T64567 CW97YT 132547287 Ki = 208 nM T64567 CW18RT 132547288 Ki = 262 nM T64567 COC54I 132547289 Ki = 133 nM T64567 CX4DM9 132547290 Ki = 85.1 nM T64567 C5JM7W 132547291 Ki = 147 nM T64567 C7V6XS 132547292 Ki = 203 nM T64567 C5O1JE 132547793 Ki > 100000 nM T64567 CKYC42 132547798 Ki > 100000 nM T64567 C7MZ8T 132569639 Ki = 180 nM T64567 CRL24F 132596304 Ki = 30.4 nM T64567 C6OA8Z 132819872 Ki = 1.7 nM T64567 CJGH58 132819873 Ki = 10.5 nM T64567 COT92G 132819874 Ki = 0.94 nM T64567 COS36W 132819875 Ki = 7 nM T64567 CMAU69 132819876 Ki = 10.5 nM T64567 CY62CQ 132938107 Ki = 1.5 nM T64567 CB8T7K 132938108 Ki = 2.7 nM T64567 CY6L7Z 132941396 Ki = 10.4 nM T64567 CD9ET2 132961426 Ki = 296 nM T64567 CR80OW 132961427 Ki = 2667 nM T64567 CEP32W 132991412 Ki = 12.1 nM T64567 C69NDK 133107891 Ki = 2.6 nM T64567 CG0HL2 134130044 Ki = 136 nM T64567 C63CQL 134130121 Ki = 1680 nM T64567 C82HUT 134130285 Ki = 918 nM T64567 CMZ76O 134130322 Ki = 172 nM T64567 C8AL2D 134130377 Ki = 1210 nM T64567 C7N0JD 134130389 Ki = 237 nM T64567 CZ7CA3 134131127 Ki = 172 nM T64567 C5XU9Y 134131319 Ki = 189 nM T64567 CZ2YK7 134131524 Ki = 1090 nM T64567 CUVB06 134131580 Ki = 306 nM T64567 C94HZF 134131659 Ki = 2.2 nM T64567 CU5B8H 134131865 Ki = 9.3 nM T64567 C2UIM6 134132835 Ki = 5.4 nM T64567 CECZ43 134133137 Ki = 20 nM T64567 C83QKJ 134133977 Ki = 18.7 nM T64567 CJ3EQ2 134136523 Ki = 16.2 nM T64567 C4IO1K 134137058 Ki = 39.8 nM T64567 CWG0L5 134139228 Ki = 20.5 nM T64567 CJ4R6E 134141819 Ki = 21.6 nM T64567 CBK73M 134146037 Ki = 14.3 nM T64567 CDH38B 134147400 Ki = 23.6 nM T64567 CDSM29 134147656 Ki = 25.4 nM T64567 C1Q8GK 134149666 Ki = 2.4 nM T64567 CF31OS 134149711 Ki = 7.5 nM T64567 C2NXB7 134151324 Ki = 10.5 nM T64567 CR4VE0 134152281 Ki = 18.4 nM T64567 CU0T4X 134152542 Ki = 2.3 nM T64567 CZ9C1N 134152694 Ki = 8.3 nM T64567 C4WBC6 134153047 Ki = 17.2 nM T64567 CSK6L9 134154625 Ki = 15.1 nM T64567 CG69UV 134155483 Ki = 24.5 nM T64567 CZ9L5F 134158397 Ki = 83.7 nM T64567 CR3Q5U 134159783 Ki = 2.2 nM T64567 CV9W6N 134159784 Ki = 2.6 nM T64567 C8C0TO 134812637 Ki = 11.4 nM T64567 CV9X5Y 134817795 Ki = 1717.9 nM T64567 C19BHQ 134817796 Ki = 262.5 nM T64567 CY3E4D 134817797 Ki = 329.5 nM T64567 C8IF6V 134817798 Ki = 23.2 nM T64567 C0UL7A 134828600 Ki = 630 nM T64567 C4ZLP6 134828601 Ki = 290 nM T64567 C3OLP6 134828602 Ki = 370 nM T64567 CJT9W0 135393499 Ki = 3.3 nM T64567 CK8FP3 135393500 Ki = 22.6 nM T64567 CRL4V7 135393501 Ki = 45.1 nM T64567 CTR37Z 135408753 Ki = 15700 nM T64567 CW9B7C 135422576 Ki = 4.5 nM T64567 C4CXD1 135434964 Ki = 15.5 nM T64567 CFK9A4 135434965 Ki = 8.3 nM T64567 CY7RT4 135442220 Ki = 780 nM T64567 CKAF26 135460193 Ki = 24 nM T64567 C0WEU9 135537166 Ki = 4.9 nM T64567 C7E8RX 135570228 IC50 = 4.53 nM T64567 CC8IO3 135595465 Ki = 190 nM T64567 C74TBX 135595467 Ki = 106 nM T64567 CX1NF7 135595474 Ki = 187 nM T64567 CL71ND 135645043 Ki > 50000 nM T64567 CHM06N 135794287 Ki = 1250 nM T64567 C1WH3Z 135891810 Ki = 8.5 nM T64567 CSH8M1 135995959 Ki = 4.3 nM T64567 CB90PQ 135995960 Ki = 4.1 nM T64567 CNG0L4 136044222 Ki = 28.1 nM T64567 CQ02AW 136044223 Ki = 251 nM T64567 C47KQP 136053622 Ki = 465 nM T64567 C1M7DN 136053656 Ki = 8.5 nM T64567 C31CEK 136094773 Ki = 8.5 nM T64567 C3VG8C 136094774 Ki = 6.4 nM T64567 C38LKD 136104491 Ki = 26000 nM T64567 C0PNH7 136104492 Ki = 7180 nM T64567 CNW21F 136104493 Ki = 7150 nM T64567 CST63W 136104494 Ki = 21000 nM T64567 C9GQS8 136104495 Ki = 9400 nM T64567 C4KH2F 136138702 Ki = 51.5 nM T64567 C4A2XS 136198631 Ki = 14.26 nM T64567 C93PWB 136198632 Ki = 24.74 nM T64567 CVME35 136198643 Ki = 295 nM T64567 CBO5I1 136242872 Ki = 9.7 nM T64567 CQDT25 136242873 Ki = 19 nM T64567 CK5AZ7 136242878 Ki = 37 nM T64567 C1NTA3 136418497 Ki = 40.1 nM T64567 C6VS7N 136607460 Ki = 3.1 nM T64567 CAC75Q 136607461 Ki = 3 nM T64567 CI28TM 136934908 Ki = 163 nM T64567 C9UKC8 136998786 Ki = 1870 nM T64567 C3QFS1 136998787 Ki = 106 nM T64567 C1P9FJ 136998788 Ki = 1880 nM T64567 CZ40LF 137028501 Ki = 8.8 nM T64567 C5Q8PD 137028502 Ki = 7.4 nM T64567 CSL47A 137028503 Ki = 20 nM T64567 C7T1HR 137028504 Ki = 4.7 nM T64567 C9WH2P 137028505 Ki = 52.9 nM T64567 CGBQ10 137028506 Ki = 9.7 nM T64567 C4DHG6 137028507 Ki = 7.8 nM T64567 CIP84X 137028508 Ki = 3.3 nM T64567 CF14KA 137028511 Ki = 15.7 nM T64567 CXHB30 137028512 Ki = 13.6 nM T64567 CRMC05 137028513 Ki = 2.8 nM T64567 CJH4E5 137028514 Ki = 2.5 nM T64567 CGAR93 137028515 Ki = 9.4 nM T64567 C4QG2K 137028516 Ki = 3.5 nM T64567 C2GMH5 137028517 Ki = 7.4 nM T64567 CBX6S7 137028518 Ki = 20 nM T64567 C52OFD 137028519 Ki = 1.1 nM T64567 CUW85H 137062187 Ki = 239 nM T64567 C4XY9S 137091066 Ki = 217 nM T64567 C64ITR 137091070 Ki = 235 nM T64567 C0BEH8 137093138 Ki = 307 nM T64567 CD6C0A 137093141 Ki = 383 nM T64567 CJ2DW1 137196867 Ki = 21.3 nM T64567 CUJ3N2 137196890 Ki = 13.3 nM T64567 CE9QV3 137226330 Ki = 6.3 nM T64567 C4SMA5 137226331 Ki = 7.7 nM T64567 C2H6VC 137226372 Ki = 192 nM T64567 CZY9D7 137226374 Ki = 240 nM T64567 C6YBD3 137226375 Ki = 5 nM T64567 C7DMR8 137226384 Ki = 14.8 nM T64567 C2KG3D 137226385 Ki = 16.7 nM T64567 C0KMB4 137226399 Ki = 194 nM T64567 CD1VC9 137226400 Ki = 208 nM T64567 C4F8NU 137226401 Ki = 237 nM T64567 CW65FQ 137226402 Ki = 201 nM T64567 CY95JF 137226420 Ki = 175 nM T64567 CM58FB 137228156 Ki = 5.8 nM T64567 CK94PV 137228157 Ki = 6.5 nM T64567 CAY48F 137228158 Ki = 7.3 nM T64567 COW81G 137273278 Ki = 34.4 nM T64567 CW52IQ 137631447 Ki = 9000 nM T64567 CRK6Y9 137631731 Ki = 261.5 nM T64567 CZ5GQ4 137631746 Ki > 100 nM T64567 C7O3CP 137632017 Ki > 50000 nM T64567 C83VZC 137632115 Ki = 160 nM T64567 CN8UL1 137632214 Ki = 8900 nM T64567 CYD0E3 137632442 Ki = 13.6 nM T64567 CH42MU 137632574 Ki = 653.7 nM T64567 CL5K3D 137632743 Ki = 28.9 nM T64567 CE20FG 137632898 Ki = 1100 nM T64567 CO25DP 137632949 Ki = 150.7 nM T64567 C9YKD5 137633039 Ki = 105.2 nM T64567 CFE79H 137633320 Ki = 277 nM T64567 CVNO32 137633860 Ki = 250.6 nM T64567 C4CIT3 137634087 Ki = 1900 nM T64567 C5NLG4 137634142 Ki = 1100 nM T64567 C7N0ER 137634525 Ki > 100000 nM T64567 C29PFJ 137634549 Ki = 1620 nM T64567 C0P6ZT 137634762 Ki = 242.4 nM T64567 CJT86I 137634882 IC50 = 152 nM T64567 C08ANJ 137635055 Ki = 330 nM T64567 CY1HI4 137635059 Ki = 76.2 nM T64567 C4YV1N 137635125 Ki = 58.1 nM T64567 C3NQ9Y 137635300 Ki = 459 nM T64567 C1ZKU2 137635320 Ki = 43.9 nM T64567 CZ1O5K 137635430 Ki = 3260 nM T64567 CS6M2N 137635469 Ki = 48.2 nM T64567 CNJV53 137635486 Ki = 8800 nM T64567 CVNX12 137635652 Ki = 54.2 nM T64567 CZ4Q1T 137636083 Ki = 13 nM T64567 C9GIX7 137636130 Ki > 50000 nM T64567 CV12YX 137636350 Ki = 31.8 nM T64567 CE46DY 137636432 Ki = 58.9 nM T64567 CK0N2Y 137636453 Ki = 22 nM T64567 CM9YC2 137636494 Ki = 18 nM T64567 CLR6U5 137636505 Ki = 428 nM T64567 C5D3BS 137636775 Ki = 350 nM T64567 CMX9T3 137636945 Ki = 7800 nM T64567 C2Z7GO 137637071 Ki = 90.9 nM T64567 CWO5Z6 137637365 Ki > 100 nM T64567 CGV9M8 137637508 Ki = 515.9 nM T64567 CG0N8K 137637564 Ki = 25.2 nM T64567 CDXW57 137637640 Ki = 2 nM T64567 CQ5K1H 137637688 Ki = 20.1 nM T64567 CPMN15 137638178 IC50 = 37 nM T64567 CB3KA0 137638304 Ki = 16.8 nM T64567 CK6OW4 137638637 Ki = 25.3 nM T64567 C6V8ED 137638882 Ki = 4.8 nM T64567 C64JQN 137639095 Ki = 9.1 nM T64567 CVJ35I 137639180 Ki = 9800 nM T64567 C12QYH 137639189 Ki = 6600 nM T64567 C4LB2X 137639339 Ki = 283.7 nM T64567 CX7TE5 137639357 Ki = 62.3 nM T64567 C0IQ1U 137639377 Ki = 677.5 nM T64567 C29XAH 137639434 Ki = 2050.6 nM T64567 CH2C3F 137639611 Ki = 20.3 nM T64567 CPR04H 137639655 Ki = 19.8 nM T64567 C95ZIL 137639751 IC50 = 20000 nM T64567 C4SP7Q 137639785 Ki = 217.9 nM T64567 COE61G 137639833 Ki = 1600 nM T64567 C5OU2V 137640459 Ki = 25.5 nM T64567 CX3JI9 137640517 Ki = 5.9 nM T64567 CZGW35 137640627 Ki = 1460 nM T64567 C8P3SC 137640892 Ki = 42.8 nM T64567 CJ4M2A 137640917 Ki = 93.1 nM T64567 CR65OQ 137640944 Ki = 42.9 nM T64567 C75WMG 137641075 Ki = 4130 nM T64567 C6B0CQ 137641198 Ki = 8.2 nM T64567 CR2MU6 137641422 Ki = 4900 nM T64567 C4FN0Q 137641666 Ki = 64.8 nM T64567 CCSN50 137642054 Ki = 20.1 nM T64567 C0Z9DH 137642233 Ki > 50000 nM T64567 C6YV7B 137642310 Ki = 380 nM T64567 CEOC90 137642331 Ki = 89.6 nM T64567 CSY67B 137642513 Ki = 319.2 nM T64567 C8Z1YM 137642848 IC50 = 60 nM T64567 C61TSP 137642864 Ki > 100000 nM T64567 C7ZX8Q 137643203 Ki = 7300 nM T64567 C1BW5I 137643671 Ki > 100000 nM T64567 CN2M3C 137643724 Ki = 990 nM T64567 C0B8QA 137643949 Ki > 100 nM T64567 CG13TO 137643998 Ki = 9100 nM T64567 CI4A9L 137644641 Ki = 3240 nM T64567 CIK49D 137644678 Ki = 21.8 nM T64567 CV75NJ 137644865 Ki = 272.6 nM T64567 CWQ91B 137644949 Ki = 45.1 nM T64567 CHG72J 137644957 Ki = 390 nM T64567 CV0AH9 137645517 Ki = 250.9 nM T64567 C6UAB5 137645654 Ki = 21.8 nM T64567 CFV6T3 137645790 Ki > 50000 nM T64567 C3CI0M 137645793 Ki = 2.4 nM T64567 CBRK83 137645944 Ki = 4.6 nM T64567 C4WOE0 137646284 Ki = 4188 nM T64567 C5WG2P 137646543 Ki = 0.5 nM T64567 C3AX0L 137647075 IC50 = 667 nM T64567 CRP78K 137647221 Ki = 54.7 nM T64567 C5T2VN 137647270 Ki = 1450 nM T64567 CXD9A0 137647636 Ki = 9 nM T64567 CY15KD 137648125 Ki = 464 nM T64567 C5PEA6 137648128 Ki = 25 nM T64567 CCD71U 137648259 Ki = 4702.5 nM T64567 CW8CL7 137648379 Ki = 80.8 nM T64567 CU81DA 137648494 Ki = 25.2 nM T64567 CK14XO 137648525 Ki = 152.6 nM T64567 C6IB1L 137648807 Ki = 38.8 nM T64567 C82NJP 137648964 Ki = 8800 nM T64567 CY94BR 137649373 Ki = 420 nM T64567 CSWR71 137649376 Ki = 93.1 nM T64567 CGLM50 137649870 Ki = 15.4 nM T64567 C2HA7Q 137649882 Ki = 64.8 nM T64567 C4N1MP 137650156 Ki = 44.5 nM T64567 CCZ4N1 137650188 Ki = 37.1 nM T64567 C1FO3T 137650198 Ki = 16.8 nM T64567 C91KQA 137650256 Ki = 4 nM T64567 CD08YK 137650293 Ki = 145.9 nM T64567 CKJ36G 137650647 Ki = 373.6 nM T64567 CD7S5L 137650698 Ki > 100000 nM T64567 CJV8Q6 137650823 Ki = 16.9 nM T64567 CBA5N4 137651134 IC50 = 95 nM T64567 C5V6XP 137651635 Ki = 4.4 nM T64567 CSTP12 137651755 Ki = 39.8 nM T64567 C01BXO 137651769 Ki = 31.3 nM T64567 CRN60L 137651808 IC50 = 33 nM T64567 CY0C6Z 137652226 Ki > 100 nM T64567 C6GWB1 137652305 Ki = 27.9 nM T64567 C5DG1K 137652445 Ki = 20.2 nM T64567 CP4GY0 137652940 Ki = 390 nM T64567 C03TAW 137653117 Ki = 250 nM T64567 CN0W6U 137653170 Ki > 50000 nM T64567 C45WNI 137653361 Ki = 9700 nM T64567 C8Y7XR 137653485 Ki = 5.8 nM T64567 CIV3E9 137653528 Ki = 3.5 nM T64567 C4U9KA 137653686 Ki > 50000 nM T64567 C0O3JI 137654169 Ki = 66.3 nM T64567 CNJ6P9 137654601 Ki = 4.6 nM T64567 CS3LD8 137654917 Ki = 190 nM T64567 CRC23M 137655132 Ki = 41 nM T64567 CWT49Q 137655252 Ki = 3850 nM T64567 C3DT7S 137655450 Ki > 100 nM T64567 CASB61 137655528 Ki = 23.5 nM T64567 C0XPN2 137655580 Ki = 639.4 nM T64567 CUO84H 137655694 Ki = 300.6 nM T64567 CAZ27T 137655913 Ki = 5.8 nM T64567 C27ALW 137655946 Ki = 7.2 nM T64567 CJV27W 137656199 IC50 = 46 nM T64567 CHD58S 137656247 Ki = 250 nM T64567 CRXD65 137656549 Ki > 50000 nM T64567 C06ONV 137656670 Ki = 20.8 nM T64567 CG5EK0 137656938 Ki = 69.5 nM T64567 CT7CW2 137657041 Ki = 1000 nM T64567 C0ME2V 137657097 Ki = 1020 nM T64567 C3PAQ7 137657121 Ki = 74.9 nM T64567 C2SYC9 137657578 Ki = 14 nM T64567 C8RNZ6 137657759 Ki > 100 nM T64567 C0KI6G 137657917 Ki = 17.9 nM T64567 CTI2V7 137658103 Ki = 26.7 nM T64567 CT5PO9 137658239 Ki = 2460 nM T64567 CH39CL 137658251 Ki = 9.5 nM T64567 C3W4BA 137658271 Ki = 113.6 nM T64567 CKX78V 137658314 Ki = 128.6 nM T64567 CL2H0T 137658375 Ki = 89.7 nM T64567 CTNZ72 137658510 IC50 = 7 nM T64567 C7V6MY 137658589 Ki = 34.5 nM T64567 CT98MV 137658877 Ki > 100 nM T64567 C8YV5D 137659052 Ki = 81.5 nM T64567 CXO9Y7 137659205 Ki = 30.8 nM T64567 CO1RD4 137659342 Ki = 330 nM T64567 C40MRZ 137659514 Ki = 10500 nM T64567 CCX48V 137659570 Ki = 261 nM T64567 C4MB7C 137659778 Ki = 45.7 nM T64567 CXK83H 137659797 Ki = 190.5 nM T64567 CHKB25 137659801 Ki = 208.2 nM T64567 CSPB10 137659919 Ki = 19.5 nM T64567 CMS92X 137660799 Ki = 25.1 nM T64567 C0TZD5 137661006 Ki > 100000 nM T64567 CQ56MJ 137661167 Ki = 287 nM T64567 C62QWK 137661307 Ki = 1471 nM T64567 CF6Z9A 137661353 Ki = 15.6 nM T64567 CRC92Y 137661359 Ki = 91.4 nM T64567 CN1JH4 137661469 Ki = 11.2 nM T64567 C1Z8KG 137661675 Ki = 36.9 nM T64567 C74YSR 137661914 Ki = 69.1 nM T64567 CO8UE3 137662293 Ki = 2782.7 nM T64567 C08ZTR 138393077 Ki = 2.6 nM T64567 CIX41M 138393379 Ki = 11.9 nM T64567 C7V9ZF 138455154 Ki = 2.8 nM T64567 CBOM51 138753317 Ki = 4.3 nM T64567 CB83JY 139593608 Ki = 1.3 nM T64567 C8TWF0 139597735 Ki = 100 nM T64567 CR10ZH 139823666 Ki > 1000 nM T64567 C78UAW 142468585 Ki = 353 nM T64567 CZY8Q6 142468589 Ki = 1.3 nM T64567 C3HMI0 142468591 Ki = 3120 nM T64567 CHA65U 142468595 Ki > 50000 nM T64567 C6KE9A 142468600 Ki > 50000 nM T64567 C65DHJ 142468602 Ki = 3300 nM T64567 CI02LX 142468604 Ki > 50000 nM T64567 C7LP3J 142468605 Ki > 50000 nM T64567 CA9O2I 142468608 Ki = 3400 nM T64567 CUE58A 142547533 Ki = 30.8 nM T64567 C6GB9T 143032987 Ki = 28.4 nM T64567 CNW7H1 145948231 Ki = 6.5 nM T64567 C3PF4Q 145948234 Ki = 6.6 nM T64567 CQC2D5 145949182 Ki = 225.1 nM T64567 C0Z2WP 145949184 Ki = 1520.4 nM T64567 CI9H2E 145949226 Ki = 77.9 nM T64567 CK65AC 145949290 Ki = 165.8 nM T64567 CP6AM5 145949377 Ki = 61.8 nM T64567 CHVR98 145949393 Ki = 11.9 nM T64567 CGLD54 145949403 Ki = 31.5 nM T64567 C3LZH7 145949437 Ki = 25.7 nM T64567 CK27DZ 145949543 IC50 = 38400 nM T64567 CROP78 145949554 Ki = 83.1 nM T64567 C09ZGW 145949615 Ki = 428.5 nM T64567 CA01QK 145949650 Ki = 1206.9 nM T64567 C7I3GC 145949670 Ki = 61.2 nM T64567 C7X0DZ 145949728 Ki = 1006 nM T64567 CIU2Y1 145949743 Ki = 217.3 nM T64567 CA05JL 145949806 Ki = 35.8 nM T64567 CHI5L3 145949836 Ki = 191 nM T64567 C3U1AB 145949909 Ki = 155.6 nM T64567 C20RXT 145949974 Ki = 10.1 nM T64567 CJS69Y 145949980 IC50 = 57310 nM T64567 CJ8R3M 145950033 Ki = 2639.1 nM T64567 CSW7B8 145950055 Ki = 90.7 nM T64567 CISR74 145950124 Ki = 227 nM T64567 CD3E6Z 145950129 IC50 = 40410 nM T64567 C5OP7G 145950184 IC50 = 6640 nM T64567 C7DBT4 145950298 Ki = 29.9 nM T64567 CO9UN4 145950340 Ki = 189.6 nM T64567 CW56LV 145950373 Ki = 0.55 nM T64567 CJSK40 145950390 Ki = 19.7 nM T64567 C2H9QY 145950512 Ki = 47.1 nM T64567 C7BK9O 145950527 Ki = 42.9 nM T64567 C63SMQ 145950568 Ki = 27.5 nM T64567 CDEJ76 145950675 IC50 = 58390 nM T64567 CE58JF 145950709 Ki = 108.4 nM T64567 C0C9FT 145950755 Ki = 8.7 nM T64567 C0AC8O 145950774 IC50 = 1840 nM T64567 C8XAH1 145950880 Ki = 7 nM T64567 C53EGH 145950894 Ki = 6 nM T64567 CRD27H 145950965 Ki = 232.3 nM T64567 C2CF0M 145950969 IC50 = 10810 nM T64567 C8IGY9 145950981 Ki = 24.2 nM T64567 C9QUL0 145951028 Ki = 2.4 nM T64567 C7W5PI 145951214 Ki = 27.3 nM T64567 C87JIM 145951255 Ki = 47.6 nM T64567 CPD05I 145951366 Ki = 2.6 nM T64567 C7LMU1 145951380 Ki = 245 nM T64567 CB8V7M 145951488 Ki = 144.4 nM T64567 CL25SI 145951508 Ki = 26.8 nM T64567 CIM8X0 145951670 Ki = 6.5 nM T64567 CH9J8K 145951685 Ki = 249.2 nM T64567 C74RDJ 145951698 Ki = 45.4 nM T64567 CJ2W6V 145951720 Ki = 2.7 nM T64567 CZ23SB 145951758 Ki = 131.5 nM T64567 CC0P1U 145951787 Ki = 1310.1 nM T64567 CF20QP 145951819 Ki = 359.6 nM T64567 C98SYV 145951855 Ki = 460.3 nM T64567 CQC79A 145951865 Ki = 126.5 nM T64567 C2OTU3 145951886 Ki = 697.4 nM T64567 CF7U3J 145951902 Ki = 79.3 nM T64567 CKZT53 145951931 Ki = 809.4 nM T64567 C3R8NQ 145951979 Ki = 3403.2 nM T64567 CGFU20 145952201 Ki = 59.4 nM T64567 C4N3QL 145952239 Ki = 8.3 nM T64567 CUJ2G6 145952345 Ki = 1.7 nM T64567 CNDQ97 145952353 IC50 = 150 nM T64567 CM30EN 145952365 Ki = 450.1 nM T64567 CU69PG 145952370 Ki = 3968.7 nM T64567 C75RDX 145952490 Ki = 2.7 nM T64567 CP92AH 145952604 Ki = 71.6 nM T64567 C26OLK 145952634 Ki = 845 nM T64567 CW42HX 145952649 Ki = 4 nM T64567 C98YOL 145952670 IC50 = 20920 nM T64567 C3ZR6A 145952729 IC50 = 57310 nM T64567 CWE6M8 145952775 Ki = 371.1 nM T64567 C81UYG 145952794 Ki = 1442 nM T64567 C6PZ3H 145952834 Ki = 136.5 nM T64567 CK4Q0X 145952846 Ki = 0.73 nM T64567 C56QVF 145952880 Ki = 5.6 nM T64567 CUB49H 145952983 Ki = 1960.4 nM T64567 CNZX07 145953044 Ki = 38.2 nM T64567 C5M0RE 145953147 IC50 = 37560 nM T64567 C5C9RI 145953173 Ki = 15.3 nM T64567 C1KQ3D 145953178 Ki = 3342.1 nM T64567 CZG27U 145953247 IC50 = 44080 nM T64567 CQM0J4 145953285 Ki = 2625.5 nM T64567 C5DJY9 145953324 Ki = 2.3 nM T64567 CZO1Y8 145953466 Ki = 324 nM T64567 CFW94A 145953493 Ki = 0.79 nM T64567 C80OQZ 145953572 Ki = 48.2 nM T64567 C7Q4IN 145953662 Ki = 44.2 nM T64567 C36ENH 145953837 Ki = 0.57 nM T64567 CH9N6D 145954010 Ki = 45.2 nM T64567 CVNE29 145954045 Ki = 1137 nM T64567 C7GIQ5 145954093 Ki = 561.2 nM T64567 CM4U3B 145954289 Ki = 39.4 nM T64567 CZE24T 145954429 IC50 = 14410 nM T64567 C7LZ1G 145954524 Ki = 39.3 nM T64567 C67HYG 145954632 Ki = 34.5 nM T64567 CZG7I4 145954697 Ki = 74.4 nM T64567 CC08PM 145954740 Ki = 361.6 nM T64567 CP80VE 145954744 IC50 = 6720 nM T64567 C0XO6A 145954770 Ki = 286.3 nM T64567 CTV8L5 145954775 Ki = 15.3 nM T64567 CNE86C 145954868 Ki = 170 nM T64567 C1LFA9 145954917 Ki = 2.4 nM T64567 CMZ2Y0 145954932 Ki = 4.8 nM T64567 CS2G9Q 145954962 IC50 = 16680 nM T64567 C0UBV8 145955012 Ki = 5.8 nM T64567 C7QL4I 145955037 Ki = 46.9 nM T64567 C6UGK8 145955158 Ki = 40 nM T64567 CM9Y2S 145955268 Ki = 91.6 nM T64567 CHTR07 145955486 Ki = 227.3 nM T64567 CS6GA9 145955537 Ki = 0.88 nM T64567 C27JZH 145955576 Ki = 127.2 nM T64567 CW90OF 145955720 Ki = 83 nM T64567 CUK18H 145955790 IC50 = 32890 nM T64567 CI64UX 145955888 Ki = 95.9 nM T64567 CB86QZ 145955914 Ki = 27.6 nM T64567 CG7W8R 145955929 Ki = 36.5 nM T64567 CDWF95 145955978 Ki = 7.5 nM T64567 C9DLX6 145955997 Ki = 46.4 nM T64567 CMGN62 145956070 Ki = 84.6 nM T64567 CS93JU 145956073 Ki = 93.1 nM T64567 CDJV68 145956076 Ki = 5.3 nM T64567 C5W1UM 145956081 Ki = 7.3 nM T64567 CHXP91 145956144 Ki = 74.7 nM T64567 CZK0L8 145956164 Ki = 22.1 nM T64567 CY1AD2 145956169 Ki = 1811.1 nM T64567 CD3LK5 145956229 Ki = 29.9 nM T64567 C89HDL 145956309 Ki = 46.4 nM T64567 CYJ3N0 145956346 Ki = 8.7 nM T64567 CQJO72 145956348 Ki = 555.2 nM T64567 CGY39T 145956363 Ki = 44.7 nM T64567 CEL63H 145956491 Ki = 104 nM T64567 CAPD95 145956503 Ki = 21.6 nM T64567 C4LH5W 145956563 Ki = 27.9 nM T64567 CRYP47 145956664 Ki = 31.5 nM T64567 CE39IU 145956732 Ki = 37.4 nM T64567 CYH7O8 145956770 Ki = 36.6 nM T64567 CWPZ94 145956803 Ki = 709.8 nM T64567 CRUI17 145956819 Ki = 107.7 nM T64567 C6I1XE 145956976 Ki = 95.4 nM T64567 C7X6NA 145957099 Ki = 37.1 nM T64567 CEF41D 145957103 Ki = 39.5 nM T64567 CAMD59 145957136 Ki = 9.3 nM T64567 C94GRZ 145957236 Ki = 0.89 nM T64567 CNLZ53 145957288 IC50 = 50920 nM T64567 CED18K 145957307 Ki = 405.2 nM T64567 CKOX92 145957394 Ki = 421.1 nM T64567 C17FUI 145957430 Ki = 248.1 nM T64567 C6OR1Q 145957438 IC50 = 130 nM T64567 CN5TM2 145957461 Ki = 1431.9 nM T64567 C4S7BR 145957546 Ki = 69.1 nM T64567 C98PXC 145957555 Ki = 383 nM T64567 CL28OB 145957582 Ki = 2805.5 nM T64567 CY37VB 145957610 IC50 = 29900 nM T64567 CP4TF7 145957664 Ki = 16.9 nM T64567 CI5B9M 145957665 Ki = 76.8 nM T64567 C6HG7S 145957711 Ki = 34.8 nM T64567 CE4O0N 145957959 Ki = 197.8 nM T64567 CXFV43 145958041 Ki = 1.9 nM T64567 C6JL8X 145958066 Ki = 41.1 nM T64567 CM07ZF 145958200 Ki = 2.7 nM T64567 CKL09Q 145958223 IC50 = 63110 nM T64567 CQO8H5 145958250 Ki = 53.6 nM T64567 CJW72B 145958328 IC50 = 44520 nM T64567 CF07KV 145958447 Ki = 47.8 nM T64567 C5URQ2 145958565 Ki = 31.6 nM T64567 CC32ZJ 145958632 Ki = 23.4 nM T64567 CQ3A6D 145958725 IC50 = 60920 nM T64567 C0PRJ7 145958803 Ki = 1659 nM T64567 CO5AK0 145958809 IC50 = 43520 nM T64567 C14UQR 145958824 Ki = 30.9 nM T64567 C2MCO8 145958917 Ki = 17 nM T64567 C0F9NS 145958940 Ki = 56.1 nM T64567 CUBA42 145958994 Ki = 39.8 nM T64567 CN69PR 145959001 IC50 = 10040 nM T64567 CNP7C0 145959116 Ki = 7 nM T64567 CU8J0M 145959118 Ki = 337.4 nM T64567 C1HML4 145959374 Ki = 1716.3 nM T64567 C37CVT 145959395 Ki = 51.3 nM T64567 C0LC9M 145959407 Ki = 439.2 nM T64567 CGK4O1 145959409 Ki = 56.3 nM T64567 CM5OK6 145959413 Ki = 43.6 nM T64567 CWNS89 145959524 Ki = 12 nM T64567 C7J6MA 145959539 Ki = 37.8 nM T64567 CJMU23 145959635 Ki = 140.7 nM T64567 CPL41Z 145959905 Ki = 15.9 nM T64567 CK8DX1 145959911 Ki = 801.2 nM T64567 CGZ1K8 145959957 Ki = 10.1 nM T64567 C29YFS 145959974 Ki = 59.2 nM T64567 CL0NM5 145960039 Ki = 418.5 nM T64567 C9MSK2 145960116 Ki = 7.4 nM T64567 CH2K1A 145960207 Ki = 79.2 nM T64567 C2SI5J 145960220 Ki = 548.6 nM T64567 CB49ZJ 145960257 Ki = 289.7 nM T64567 C6JND4 145960287 Ki = 2.4 nM T64567 C3JTG4 145960436 Ki = 378 nM T64567 C89GHI 145960779 Ki = 177 nM T64567 CVMF36 145960835 Ki = 373 nM T64567 CBGV25 145960853 Ki = 143 nM T64567 CT6U2G 145961010 Ki = 1589.1 nM T64567 CD2X3F 145961133 Ki = 24.2 nM T64567 CBT85V 145961452 Ki = 43.6 nM T64567 C6JG2V 145961631 Ki = 2.4 nM T64567 CDA7G0 145962071 Ki = 205 nM T64567 CCYK28 145962259 Ki = 502 nM T64567 CQV18P 145962416 Ki = 502 nM T64567 C14OZY 145962693 Ki = 166.1 nM T64567 C34BRN 145962803 Ki = 430 nM T64567 C36LCF 145962935 Ki = 16.5 nM T64567 CZ9PL4 145963030 Ki = 33.1 nM T64567 C0CP9O 145963122 IC50 = 40180 nM T64567 CGY68S 145963294 Ki = 489 nM T64567 CJU15K 145963586 Ki = 44.3 nM T64567 CVL39I 145963679 Ki = 468 nM T64567 CUZ3A5 145963719 Ki = 159 nM T64567 C5VI0K 145964063 Ki = 8.7 nM T64567 CM71JT 145964104 Ki = 59.9 nM T64567 CGTA80 145964130 Ki = 45.5 nM T64567 C9DE8Y 145964275 Ki = 15.9 nM T64567 C4C9IE 145964340 Ki = 26.2 nM T64567 CK21BE 145964400 Ki = 144.4 nM T64567 CAPU84 145964558 Ki = 8 nM T64567 C6FE1K 145964671 Ki = 54.9 nM T64567 CTC21S 145964779 Ki = 329.7 nM T64567 C3F4IS 145965133 Ki = 26.6 nM T64567 CGR16W 145965551 Ki = 7360 nM T64567 C6RZT2 145965743 Ki = 123.3 nM T64567 CWHV36 145965762 Ki = 3020 nM T64567 CINP09 145966173 Ki = 90.6 nM T64567 C2G8VU 145966250 Ki = 63 nM T64567 C5X7FM 145966343 Ki = 169.8 nM T64567 CCDI76 145966475 Ki = 10.4 nM T64567 CMF72D 145966553 Ki = 56.1 nM T64567 CQ64RX 145966558 Ki = 141 nM T64567 CJ4D0R 145967030 Ki = 244.4 nM T64567 C7SUX3 145967040 Ki = 137.1 nM T64567 C7HZ6V 145967049 Ki = 62.4 nM T64567 CP8Q9U 145967308 Ki = 72.1 nM T64567 CFY3M6 145968026 Ki = 93.1 nM T64567 CDYR51 145968242 Ki = 51.9 nM T64567 C10PQH 145968245 Ki = 4.8 nM T64567 CKME70 145968701 Ki = 21.2 nM T64567 CX4D2R 145969379 Ki = 18.3 nM T64567 C9R4VB 145971458 Ki = 182.1 nM T64567 CD9I1U 145971467 Ki = 2.4 nM T64567 CZ71HS 145971486 Ki = 38.1 nM T64567 CC8D6E 145971537 IC50 = 26150 nM T64567 C73WMA 145971736 Ki = 145.2 nM T64567 C9P6UE 145971793 Ki = 15.9 nM T64567 C6DQK4 145972104 Ki = 16.3 nM T64567 CO4V1G 145972192 Ki = 181.1 nM T64567 CYMF38 145972316 Ki = 17.5 nM T64567 CP9H1U 145972366 Ki = 146.3 nM T64567 CD42QZ 145972397 Ki = 5.1 nM T64567 C93LTU 145972477 IC50 = 150 nM T64567 CZ2LP7 145972551 Ki = 66.6 nM T64567 COJ6K4 145972603 Ki = 34.1 nM T64567 CS6D5R 145972711 IC50 = 1610 nM T64567 CGE23X 145972719 Ki = 1071 nM T64567 CFXW14 145972912 Ki = 93 nM T64567 CF5KR4 145972986 Ki = 7.7 nM T64567 C65ZVF 145973004 Ki = 24.7 nM T64567 CN20BQ 145973308 Ki = 321.1 nM T64567 C1I8GK 145973355 Ki = 112.7 nM T64567 C9MZS1 145973465 Ki = 103.2 nM T64567 C8UAD6 145973595 Ki = 17.8 nM T64567 C7Y3WO 145973882 Ki = 3.9 nM T64567 C2C1KE 145973952 Ki = 117.5 nM T64567 CJ15WQ 145974101 Ki = 5.2 nM T64567 C7ZRI0 145974266 Ki = 47 nM T64567 CX5U8J 145974401 Ki = 12.5 nM T64567 CJD0I1 145974412 Ki = 4510 nM T64567 C2MF3Y 145974672 Ki = 5.8 nM T64567 C1QZ7F 145974710 Ki = 62.5 nM T64567 CG5SL1 145974949 Ki = 97.8 nM T64567 CVPA83 145974992 Ki = 5.8 nM T64567 CDU4M5 145975077 Ki = 76.5 nM T64567 C3I2WU 145975151 Ki = 43.3 nM T64567 C5U8RK 145975281 Ki = 62 nM T64567 C1VJD3 145975355 Ki = 100.1 nM T64567 CBL8Y4 145975424 Ki = 22 nM T64567 CT16KB 145975591 Ki = 4.8 nM T64567 CPK17Y 145975721 Ki = 7900 nM T64567 CZVK21 145975933 Ki = 72.2 nM T64567 CQ08AT 145976207 Ki = 1206.9 nM T64567 CO9M3B 145976300 Ki = 18900 nM T64567 CI9C6U 145976539 Ki = 38.1 nM T64567 CZ7QU1 145976656 Ki = 3.1 nM T64567 C2BIZ4 145976658 Ki = 38.9 nM T64567 CHI26Q 145976735 Ki = 94.9 nM T64567 CZWC63 145977536 Ki = 177.2 nM T64567 CH3IC0 145977574 Ki = 23.1 nM T64567 CUEB47 145977814 Ki = 61.3 nM T64567 C81JIQ 145977869 Ki = 78.9 nM T64567 CL7GH8 145977904 Ki = 16.1 nM T64567 CK9L7E 145977947 Ki = 39.5 nM T64567 C69UQY 145978025 Ki = 202.4 nM T64567 C5QSK0 145978140 Ki = 17.7 nM T64567 CO0J6L 145978583 Ki = 172 nM T64567 CYG69V 145978605 Ki = 39.3 nM T64567 CYWK54 145978673 Ki = 14 nM T64567 C2D1TO 145978690 Ki = 48 nM T64567 CA32BT 145978780 Ki = 18.3 nM T64567 CXI41R 145978938 Ki = 170 nM T64567 CM8KP7 145979094 Ki = 340 nM T64567 C82LKO 145979169 Ki = 240 nM T64567 CI34JB 145979332 Ki = 77.9 nM T64567 CSPH69 145979414 Ki = 1631.4 nM T64567 CQDB02 145979430 Ki = 1272.6 nM T64567 CUDO01 145979473 Ki = 235.3 nM T64567 COYX31 145979594 Ki = 134.1 nM T64567 CFUC92 145979600 Ki = 9 nM T64567 CXDE63 145979618 Ki = 2260 nM T64567 C7ZOM8 145979619 Ki = 3430 nM T64567 CIF72X 145979737 Ki = 151.5 nM T64567 CMT6G7 145979772 Ki = 81.2 nM T64567 C8YA0B 145979831 Ki = 0.87 nM T64567 C5S9JX 145979949 Ki = 7.1 nM T64567 C9H6AW 145979979 Ki = 2780 nM T64567 CLFJ74 145980146 Ki = 1788.6 nM T64567 CD1IJ2 145980204 Ki = 9.1 nM T64567 CS85AP 145980216 Ki = 2250 nM T64567 CWA24U 145980366 Ki = 101.2 nM T64567 CE3DP8 145980765 Ki = 7 nM T64567 C85TGI 145980938 Ki = 17.7 nM T64567 C97LPB 145981035 Ki = 31.5 nM T64567 C1RO4L 145981799 Ki = 100 nM T64567 C15PEL 145982039 Ki = 7.5 nM T64567 C4DNF7 145982126 Ki = 177.2 nM T64567 C7N6RT 145982437 Ki = 12.3 nM T64567 C2O8PK 145982576 Ki = 256.4 nM T64567 CK8MY4 145982622 Ki = 107.2 nM T64567 CX6Y5G 145982786 Ki = 737.7 nM T64567 C7M0HW 145982836 Ki = 1477 nM T64567 C34LIQ 145982969 Ki = 1307 nM T64567 CH3EF7 145983056 Ki = 1406 nM T64567 CN7G5J 145983107 Ki = 2089 nM T64567 C90VNX 145983131 Ki = 2333 nM T64567 C9S0WG 145983404 Ki = 1841 nM T64567 CWUJ59 145983568 Ki = 633 nM T64567 CB5G4W 145983664 Ki = 95.2 nM T64567 CF26VG 145983797 Ki = 2905 nM T64567 C5SLN9 145983850 Ki = 909 nM T64567 CI52KO 145983856 Ki = 2373 nM T64567 C3J5NQ 145983899 Ki = 264.5 nM T64567 C8PM9Y 145984067 Ki = 73 nM T64567 CA6I9T 145984095 Ki = 227.5 nM T64567 CEA52W 145984222 Ki = 1353 nM T64567 CO9P3M 145984354 Ki = 2833 nM T64567 C49ALP 145984517 Ki = 1730 nM T64567 C8C0AB 145984626 Ki = 1931.7 nM T64567 CLDZ58 145984801 Ki = 715.5 nM T64567 C05FCU 145984802 Ki = 71.2 nM T64567 C7N6ZB 145984855 Ki = 1581 nM T64567 C4FBS2 145985005 Ki = 1415 nM T64567 CZ8NA9 145985353 Ki = 1213 nM T64567 C8Y1UT 145985534 Ki = 198.3 nM T64567 CF16KP 145985651 Ki = 8.2 nM T64567 CJEG52 145985679 Ki = 237.2 nM T64567 CN1WK4 145985761 Ki = 730.3 nM T64567 CIT98E 145985912 Ki = 1423 nM T64567 C8VIF2 145985922 Ki = 225.4 nM T64567 CX0YW6 145985969 Ki = 2451 nM T64567 C3E0RD 145986123 Ki = 14.3 nM T64567 CF7CH8 145986297 Ki = 116.7 nM T64567 CTZ71U 145986436 Ki = 340 nM T64567 CIDO62 145986509 Ki = 530 nM T64567 CK05FT 145986641 Ki = 110 nM T64567 CN56XE 145986933 Ki = 1853.6 nM T64567 CG6CU5 145987209 Ki = 231.4 nM T64567 CT01AM 145987366 Ki = 150 nM T64567 C9UBE8 145987408 Ki = 0.55 nM T64567 CZPA17 145987454 Ki = 30.4 nM T64567 CI9F3V 145987533 Ki = 30.1 nM T64567 C65QOW 145987697 Ki = 6.5 nM T64567 CQF4O8 145987804 Ki = 148.3 nM T64567 CBF3V2 145987828 Ki = 26.3 nM T64567 C0LVN9 145987839 Ki = 715.6 nM T64567 C6RMF1 145987996 Ki = 0.89 nM T64567 C8XDH5 145988129 Ki = 390 nM T64567 C89RFU 145988368 Ki = 7.2 nM T64567 CJ1P5W 145988462 Ki = 2491.8 nM T64567 CXA6F3 145988572 Ki = 7.6 nM T64567 CO3N6M 145988784 Ki = 157 nM T64567 CPZN93 145988792 Ki = 27.4 nM T64567 CZW72V 145988876 Ki = 254.1 nM T64567 C1LV0U 145988936 Ki = 2231.8 nM T64567 C39ZMI 145988963 Ki = 14.2 nM T64567 C7AUF1 145989028 Ki = 31 nM T64567 C6BKP8 145989063 Ki = 90 nM T64567 C35VEG 145989087 Ki = 2440 nM T64567 C6DN9E 145989219 Ki = 1250 nM T64567 COZM89 145989422 Ki = 130 nM T64567 CJH51I 145989433 Ki = 3540 nM T64567 C9RVK0 145989853 Ki = 1660.9 nM T64567 CYJ79A 145989992 Ki = 2.6 nM T64567 CA8K2J 145990039 Ki = 30.6 nM T64567 C8XD2V 145990044 Ki = 940 nM T64567 CLQ12A 145990129 Ki = 23.6 nM T64567 CHMR39 145990191 Ki = 162.7 nM T64567 CYOD69 145990290 Ki = 1243.6 nM T64567 CZB2X3 145990392 Ki = 1903.1 nM T64567 CB63XC 145990519 Ki = 275.7 nM T64567 CJQ73W 145990589 Ki = 196.9 nM T64567 C2WTN6 145990640 Ki = 25.2 nM T64567 CM6SA4 145990881 Ki = 169 nM T64567 CIA37P 145991377 Ki = 2.9 nM T64567 CWH89P 145991839 Ki = 13.9 nM T64567 C3QXL4 145991981 Ki = 1046.3 nM T64567 C9F8TL 145992666 Ki = 6.9 nM T64567 C58FGU 145992776 Ki = 150 nM T64567 C7RYJ4 145992796 Ki = 1956.6 nM T64567 CE34YK 145992956 Ki = 1738.1 nM T64567 CH48GI 145992962 Ki = 205.6 nM T64567 CO42RK 145992983 Ki = 23.8 nM T64567 C8IE2X 145993014 Ki = 32.3 nM T64567 CDC84X 145993019 Ki = 25.8 nM T64567 C7OZD6 145993265 Ki = 56.3 nM T64567 CE0HY6 145993300 Ki = 19.9 nM T64567 CS40WA 145993323 Ki = 8.4 nM T64567 CMS86X 145993352 Ki = 290 nM T64567 CB12JK 145993432 Ki = 179.7 nM T64567 CZSC36 145993499 Ki = 8.9 nM T64567 CEC07M 145993642 Ki = 460 nM T64567 CK3YT9 145993866 Ki = 5.4 nM T64567 CIDP76 145994238 Ki = 2.6 nM T64567 C48CZD 146160385 Ki = 26.1 nM T64567 C2SG4L 146833326 Ki = 45.5 nM T64567 C6FD2N 147348395 Ki = 88.1 nM T64567 CGMX98 155510724 Ki = 4.6 nM T64567 C06MEW 155510831 Ki = 192 nM T64567 C3QJI5 155510851 Ki = 0.46 nM T64567 CY5T1K 155510897 Ki = 1186 nM T64567 C1PG9M 155511036 Ki = 118.1 nM T64567 CN6DW9 155511075 Ki = 12.1 nM T64567 C2PXC3 155511133 Ki = 3.8 nM T64567 C1A5OB 155511232 Ki = 46.3 nM T64567 C30ADE 155511364 Ki = 169.2 nM T64567 C1D8JF 155511459 Ki = 132.7 nM T64567 C6QNX5 155511723 Ki = 15.2 nM T64567 C03BJU 155511800 Ki = 520 nM T64567 CJA94W 155512108 Ki = 9.5 nM T64567 CMCL94 155512138 Ki = 13.1 nM T64567 CI40CL 155512225 Ki = 41.3 nM T64567 C1ZPW3 155512418 Ki = 177.2 nM T64567 CQC04P 155512706 Ki = 204.4 nM T64567 C7J0HP 155512942 Ki = 96500 nM T64567 C51PHM 155512962 Ki = 347.3 nM T64567 CN53ED 155512974 Ki = 96700 nM T64567 CLX19M 155512982 Ki = 242.8 nM T64567 CVSG61 155513076 Ki = 89.5 nM T64567 C21CAW 155513169 Ki = 1240.4 nM T64567 CW1DP7 155513481 Ki = 6.9 nM T64567 C7QT4V 155513609 Ki > 10000 nM T64567 C5VT4X 155514082 Ki = 17.6 nM T64567 CX2UJ9 155514131 Ki = 4500 nM T64567 CV7WR4 155514243 Ki = 37.9 nM T64567 C67VGD 155514389 Ki = 0.88 nM T64567 C7W9NI 155514825 Ki = 5400 nM T64567 CU9H2A 155514935 Ki = 40.2 nM T64567 CMQV46 155514970 Ki = 7.1 nM T64567 CR89MP 155515069 Ki = 0.7 nM T64567 CCQB03 155515285 Ki = 333.2 nM T64567 CW08ZX 155515305 Ki = 530 nM T64567 C5IPM8 155515308 Ki = 86.2 nM T64567 C46UNX 155515514 Ki = 8.6 nM T64567 C6DG3E 155515525 Ki > 100000 nM T64567 C7MER6 155515557 Ki = 460 nM T64567 C7UQ3J 155515746 Ki = 942 nM T64567 CT2ZB0 155515980 Ki = 24.9 nM T64567 C74SEH 155516204 Ki > 100000 nM T64567 CM9F7H 155516281 Ki > 50000 nM T64567 CLNT85 155516404 Ki = 6.5 nM T64567 COP4Q6 155516517 Ki = 104.7 nM T64567 C9LWV6 155516550 Ki = 10.5 nM T64567 C7IR3P 155516553 Ki = 6800 nM T64567 CBV6D3 155516701 Ki = 23.7 nM T64567 CP0NH3 155516885 Ki = 1166 nM T64567 CAG9L4 155517430 Ki = 93 nM T64567 C3OW4N 155517544 Ki > 50000 nM T64567 CW18JG 155517622 Ki = 150.7 nM T64567 C2H3JR 155517687 Ki > 100000 nM T64567 CQI20B 155517798 Ki = 8200 nM T64567 CRP2A6 155517861 Ki = 29.4 nM T64567 CWP3G6 155517862 Ki = 195.9 nM T64567 CHA2R1 155517933 Ki = 277.9 nM T64567 CF07ZS 155517996 Ki = 32.8 nM T64567 C0O5CN 155518098 Ki = 157.9 nM T64567 CUN49T 155518138 Ki = 4.9 nM T64567 C92QDE 155518180 Ki = 58.9 nM T64567 C1VNX3 155518220 Ki = 13.2 nM T64567 CP0U8D 155518225 Ki > 50000 nM T64567 CP7UI1 155518510 Ki = 17.5 nM T64567 CM7DQ6 155518807 Ki = 226.3 nM T64567 CHI59Y 155518875 Ki = 94900 nM T64567 CL92UI 155519026 Ki = 10.1 nM T64567 C5TO4Q 155519047 Ki > 100000 nM T64567 CRF95N 155519064 Ki = 184.8 nM T64567 CN8RC2 155519138 Ki = 4600 nM T64567 CK21TJ 155519240 Ki = 9.4 nM T64567 C8MYG2 155519248 Ki = 22.6 nM T64567 CO6D1Y 155519288 Ki = 27 nM T64567 CT56OD 155519473 Ki = 7.2 nM T64567 CI18TP 155519626 Ki = 45.5 nM T64567 CP4IL9 155519983 Ki = 20.9 nM T64567 CIV68R 155520019 Ki = 18.7 nM T64567 C5PN0D 155520029 Ki = 245.4 nM T64567 CP49HE 155520274 Ki = 17.8 nM T64567 C4Z8MX 155520314 Ki = 11.8 nM T64567 C5JCL6 155520507 Ki = 474.3 nM T64567 CG4VJ8 155520652 Ki = 12600 nM T64567 C8E0SN 155520671 Ki = 6600 nM T64567 CE8QY5 155520792 Ki = 476.5 nM T64567 C80OQU 155520908 Ki > 50000 nM T64567 CQ0OR1 155520930 Ki = 1588.1 nM T64567 CBM47H 155520952 Ki = 17.6 nM T64567 C9Z1FL 155521038 Ki = 100.6 nM T64567 C2J1YG 155521041 Ki = 2.6 nM T64567 C2PR8W 155521294 Ki = 273.8 nM T64567 CN2X1Q 155521353 Ki = 8.8 nM T64567 CB54YX 155521489 Ki = 3.3 nM T64567 CRQ4L3 155521766 Ki = 15.5 nM T64567 CNP87G 155521876 Ki = 55.8 nM T64567 CR49AJ 155521885 Ki = 2.3 nM T64567 C4IYX7 155521930 Ki = 36.9 nM T64567 C2Q7BG 155522085 Ki = 63.6 nM T64567 C0A4EO 155522100 Ki = 16.7 nM T64567 CSN4C2 155522321 Ki = 51.1 nM T64567 C70NUX 155522372 Ki = 73.2 nM T64567 C8K9OI 155522618 Ki = 1.6 nM T64567 CDN9Z5 155522816 Ki = 28.2 nM T64567 C0Z3QT 155522883 Ki = 42 nM T64567 CJ49ZN 155522995 Ki = 49.9 nM T64567 C3HGK6 155523328 Ki = 19.6 nM T64567 C6YZM3 155523403 Ki > 100 nM T64567 C9Q2WR 155523406 Ki = 14.1 nM T64567 CU2N9J 155523547 Ki = 5.9 nM T64567 CIF91M 155523572 Ki = 0.77 nM T64567 C8WP5K 155523621 Ki = 21.1 nM T64567 C9LF7B 155523634 Ki > 100000 nM T64567 C4U8XN 155523810 Ki = 13.8 nM T64567 CWD9Y1 155523853 Ki = 3.1 nM T64567 C3MX7F 155523857 Ki = 293.9 nM T64567 C0MZ5G 155524206 Ki = 0.6 nM T64567 C6KCG7 155524248 Ki > 50000 nM T64567 CSC58M 155524279 Ki = 3412.4 nM T64567 CK86ZT 155524367 Ki = 15 nM T64567 CK80AQ 155524610 Ki = 43.6 nM T64567 C9PV5X 155524649 Ki > 100000 nM T64567 CDO4X2 155524724 Ki = 41.1 nM T64567 C3DM5L 155524759 Ki = 187.5 nM T64567 C5J8AS 155524785 Ki = 19.6 nM T64567 CS0WP1 155524852 Ki = 18430 nM T64567 C8M1KI 155525036 Ki = 28.6 nM T64567 CV6N0C 155525231 Ki = 15.3 nM T64567 CHT29F 155525313 Ki = 105.3 nM T64567 CPL80N 155525961 Ki = 17.6 nM T64567 C4R1OT 155526288 Ki = 1186 nM T64567 CGC8Y0 155526420 Ki = 273.5 nM T64567 CKT14B 155526554 Ki = 47.7 nM T64567 C0XZD3 155526695 Ki > 50000 nM T64567 CWGS97 155526825 Ki = 74 nM T64567 CGV91K 155527018 Ki = 43.3 nM T64567 CCL7V8 155527060 Ki = 38.1 nM T64567 CNVX86 155527078 Ki = 35.9 nM T64567 CG8JZ9 155527153 Ki = 34.4 nM T64567 C8K3OI 155527167 Ki = 5.2 nM T64567 C1LDV0 155527209 Ki = 19.7 nM T64567 C1I5PO 155527240 Ki > 50000 nM T64567 CK8XN6 155527284 Ki = 127.5 nM T64567 C4N7OY 155527400 Ki = 15.9 nM T64567 CJ3K9W 155527428 Ki = 25.1 nM T64567 C4A5BC 155527483 Ki = 25.5 nM T64567 C7YW9E 155527622 Ki > 50000 nM T64567 C65FOA 155527703 Ki = 36.9 nM T64567 C07LVI 155527781 Ki = 19.4 nM T64567 CPAH30 155527788 Ki = 9.2 nM T64567 C5XC7V 155527967 Ki = 2028 nM T64567 C0RJ2M 155528294 Ki = 33 nM T64567 CN9G0E 155528332 Ki = 223 nM T64567 C4IML7 155528345 Ki = 46.8 nM T64567 CB08MU 155528753 Ki > 100000 nM T64567 C5X0CS 155528825 Ki > 100000 nM T64567 CN27OU 155528858 Ki = 3298 nM T64567 C7DCG0 155529026 Ki = 15.9 nM T64567 CECZ45 155529036 Ki = 188.3 nM T64567 C1T2EA 155529101 Ki = 6.6 nM T64567 CWEQ38 155529122 Ki = 27.9 nM T64567 C52QUD 155529352 Ki = 7.6 nM T64567 CG94RZ 155529376 Ki = 87.9 nM T64567 C2NY1E 155529877 Ki = 4.9 nM T64567 C2JV7R 155529885 Ki = 680 nM T64567 CJ21OD 155530289 Ki > 50000 nM T64567 CW07EO 155530326 Ki = 51 nM T64567 CKO2V5 155530358 Ki = 47.2 nM T64567 C7TV5H 155530408 Ki = 94 nM T64567 C9Y4VC 155530502 Ki = 0.62 nM T64567 CTJ3I7 155530506 Ki = 6.4 nM T64567 C0HQ8E 155530537 Ki = 3.7 nM T64567 CP3UJ0 155530687 Ki = 0.31 nM T64567 C2T0LQ 155530848 Ki = 22.1 nM T64567 C3GK9H 155530900 Ki = 48.7 nM T64567 C2MT3K 155530925 Ki = 49 nM T64567 C2X1JQ 155530996 Ki = 1.4 nM T64567 COY7L3 155531072 Ki = 15.9 nM T64567 C8C4BT 155531090 Ki > 50000 nM T64567 CICU68 155531183 Ki = 8.8 nM T64567 CGN43T 155531186 Ki = 6.2 nM T64567 CO7P5W 155531268 Ki = 18.4 nM T64567 CLMZ93 155531382 Ki = 28.9 nM T64567 CYBD02 155531537 Ki = 4872 nM T64567 C43LZI 155531630 Ki = 8.2 nM T64567 CC5L6V 155531813 Ki = 7.7 nM T64567 CFV23M 155531820 Ki > 100000 nM T64567 CW6TC5 155531936 Ki = 2100 nM T64567 C03TYX 155531975 Ki = 35.1 nM T64567 CUM2B8 155532026 Ki = 54700 nM T64567 C83DJY 155532441 Ki = 47300 nM T64567 CASV53 155532466 Ki = 26.7 nM T64567 CFK8R5 155532512 Ki > 100000 nM T64567 CQ0XM6 155532587 Ki = 43.3 nM T64567 C5H8QF 155532861 Ki = 30.2 nM T64567 CG7Y5M 155532951 Ki = 450 nM T64567 CKY1I8 155533416 Ki = 89.6 nM T64567 CDM2Y1 155533454 Ki = 1.8 nM T64567 C64XYO 155533459 Ki = 2.4 nM T64567 CPX2T1 155533590 Ki = 4.3 nM T64567 COK37H 155533887 Ki > 50000 nM T64567 CTKI39 155533898 Ki = 2828.4 nM T64567 C0I5XS 155534055 Ki > 50000 nM T64567 C78ZFI 155534074 Ki = 7.8 nM T64567 CT5NG1 155534179 Ki = 3.3 nM T64567 CPG13Y 155534247 Ki = 7.8 nM T64567 C6UF3R 155534332 Ki = 26.4 nM T64567 CR2A6J 155534340 Ki = 205 nM T64567 C14TGQ 155534675 Ki = 6.9 nM T64567 CK4TR2 155534861 Ki = 102.9 nM T64567 CS5OI9 155534862 Ki = 92.4 nM T64567 CHG10E 155534912 Ki = 2.8 nM T64567 C67ROE 155534951 Ki = 17.6 nM T64567 CE1I8S 155535343 Ki = 31.5 nM T64567 CC7M4N 155535347 Ki = 1088 nM T64567 CVU5P6 155535355 Ki = 2.6 nM T64567 CV0N9I 155535382 Ki = 2254.4 nM T64567 CNFR72 155535756 Ki > 100000 nM T64567 CD2O3A 155535852 Ki = 543 nM T64567 CLJ64Q 155535889 Ki = 8.4 nM T64567 CZPY79 155536184 Ki = 4.2 nM T64567 CF0PC4 155536422 Ki = 247.1 nM T64567 CW92OP 155536652 Ki = 22.4 nM T64567 CB47KF 155536691 Ki = 26.4 nM T64567 CZ0T6A 155537018 Ki = 60.2 nM T64567 C6T7BQ 155537167 Ki = 2967 nM T64567 C1K9AC 155537404 Ki = 192 nM T64567 CXQ23T 155537493 Ki > 100000 nM T64567 C4K0MB 155537772 Ki > 100000 nM T64567 C0CG6Q 155537790 Ki = 25.8 nM T64567 C47OHJ 155537809 Ki = 7.3 nM T64567 C67ZET 155537843 Ki = 19.2 nM T64567 C60IZQ 155538189 Ki = 231 nM T64567 CB2EI4 155538212 Ki = 18.3 nM T64567 C9AP8F 155538224 Ki = 3.2 nM T64567 CB8C4X 155538289 Ki = 5400 nM T64567 C3XSM6 155538611 Ki = 2184 nM T64567 CM6D1H 155538676 Ki = 189.8 nM T64567 CHQP36 155539441 Ki = 9.4 nM T64567 CKE72Y 155539552 Ki = 2.2 nM T64567 C94OZU 155539579 Ki = 81.2 nM T64567 CS1G5V 155539783 Ki = 25 nM T64567 C53TKA 155540088 Ki = 11.8 nM T64567 CSAD81 155540401 Ki = 19.5 nM T64567 CW9B0X 155540441 Ki = 133 nM T64567 C2VAD8 155540596 Ki = 1.1 nM T64567 C95TBC 155540629 Ki = 5680 nM T64567 CCO34J 155540665 Ki = 230.2 nM T64567 CGNS87 155540756 Ki = 2.1 nM T64567 CFN03K 155540920 Ki = 21.6 nM T64567 C4H1ZC 155541040 Ki = 7.8 nM T64567 C3CLU2 155541078 Ki = 13.5 nM T64567 C7Z6FC 155541724 Ki = 6187.6 nM T64567 C8RV6T 155541805 Ki = 3.5 nM T64567 CW96ES 155541807 Ki = 10.5 nM T64567 C5F3SJ 155541888 Ki = 7.7 nM T64567 CX20DK 155541945 Ki = 1480 nM T64567 CA46FW 155542038 Ki = 17.3 nM T64567 CZ2CT0 155542259 Ki = 233 nM T64567 CA75HO 155542580 Ki = 41.3 nM T64567 CTL8O3 155542606 Ki = 14 nM T64567 C3RC8T 155542635 Ki = 16.5 nM T64567 CA76LB 155542698 Ki = 720 nM T64567 CY3BO6 155542934 Ki = 3016.3 nM T64567 C75TVG 155542954 Ki = 6.4 nM T64567 C2AEH6 155543096 Ki = 539 nM T64567 CHKV89 155543295 Ki = 0.39 nM T64567 CRF64E 155543422 Ki = 2 nM T64567 CLF3N5 155543891 Ki = 0.7 nM T64567 CPV20B 155543950 Ki = 11.2 nM T64567 C08DHT 155544006 Ki = 189.5 nM T64567 C30HST 155544165 Ki = 45.1 nM T64567 CN0E1V 155544321 Ki = 9.2 nM T64567 CS9WR6 155544336 Ki = 11.7 nM T64567 C7PC5J 155544382 Ki = 0.24 nM T64567 CSX2H7 155544608 Ki = 47.9 nM T64567 CRM69J 155544710 Ki = 25 nM T64567 CP27AW 155544846 Ki = 40.3 nM T64567 CDXL09 155544901 Ki = 3.5 nM T64567 C0BV1J 155545536 Ki = 7.3 nM T64567 CQV78W 155545657 Ki = 3.3 nM T64567 CB6J9G 155545674 Ki = 136.6 nM T64567 CY6SX5 155545800 Ki = 38600 nM T64567 CP2SZ7 155545812 Ki > 50000 nM T64567 C95IJM 155545916 Ki = 312 nM T64567 C3Y8LT 155546146 Ki = 17.6 nM T64567 C5MTW6 155546162 Ki = 9.7 nM T64567 CSW62L 155546892 Ki = 8629 nM T64567 CC4IG8 155547081 Ki = 17.6 nM T64567 CF3UL5 155547275 Ki = 22.8 nM T64567 CV7OB5 155547342 Ki > 100000 nM T64567 C9E2KH 155547486 Ki = 4.7 nM T64567 C59MDT 155547507 Ki = 22.8 nM T64567 C83ZIS 155547526 Ki = 16.2 nM T64567 CW19PC 155547551 Ki = 67.9 nM T64567 C73YLV 155547628 Ki = 808.9 nM T64567 C9FVY6 155547723 Ki = 8.3 nM T64567 C61MSB 155547730 Ki = 14.8 nM T64567 CK5UD3 155547819 Ki = 33.4 nM T64567 CU94YA 155548070 Ki = 21.5 nM T64567 CCUN29 155548118 Ki = 16 nM T64567 C3IO2B 155548134 Ki = 48.6 nM T64567 C3JYG2 155548272 Ki = 28.6 nM T64567 CQG5F9 155548326 Ki = 6.6 nM T64567 C6XBZ3 155548352 Ki = 27.3 nM T64567 CUTY40 155548640 Ki = 8.2 nM T64567 CALV26 155548675 Ki = 0.16 nM T64567 CH2KB7 155548697 Ki = 3.7 nM T64567 CN7S5W 155548866 Ki = 16.4 nM T64567 CDC0F4 155548911 Ki = 176.7 nM T64567 CU1NE7 155549031 Ki = 476.6 nM T64567 C9JOV3 155549090 Ki = 22.4 nM T64567 CR79SY 155549354 Ki = 27.2 nM T64567 CL2B4T 155549378 Ki = 8.9 nM T64567 C6PY2G 155549478 Ki = 3.5 nM T64567 C2CLU0 155549558 Ki = 31.5 nM T64567 CIG6A7 155549616 Ki = 2450 nM T64567 C1JR2F 155549662 Ki = 230.5 nM T64567 CF6CW3 155549677 Ki = 66.9 nM T64567 C8NS5F 155549723 Ki = 280 nM T64567 CEZX49 155549753 Ki = 34.1 nM T64567 C8GZK4 155549788 Ki > 100000 nM T64567 CAYO49 155550021 Ki = 0.81 nM T64567 C3YN0W 155550099 Ki = 2967.4 nM T64567 CZB57Y 155550558 Ki = 0.49 nM T64567 CHO96B 155550610 Ki = 960 nM T64567 C4O6TN 155550616 Ki = 61.9 nM T64567 CMWQ79 155550618 Ki = 1.8 nM T64567 CB2Q4M 155550927 Ki = 9.7 nM T64567 CG0MQ3 155551020 Ki = 0.58 nM T64567 CTE04H 155551088 Ki = 203 nM T64567 C4S0JZ 155551334 Ki = 51.2 nM T64567 CL2H8V 155551536 Ki > 100000 nM T64567 CSY39H 155551651 Ki = 2510 nM T64567 C69AYQ 155551705 Ki > 100000 nM T64567 COC4Z9 155551784 Ki = 20.9 nM T64567 CZ0T3C 155551786 Ki = 0.8 nM T64567 C3AN2K 155551935 Ki = 1120 nM T64567 C7E3UF 155552316 Ki = 8000 nM T64567 C3DHB7 155552411 Ki > 50000 nM T64567 CZ6VL4 155552603 Ki = 17.6 nM T64567 CN25FV 155552708 Ki = 2.4 nM T64567 CBQ42J 155552773 Ki = 5200 nM T64567 CFT82G 155552780 Ki = 86.1 nM T64567 C0OG8P 155553361 Ki = 0.13 nM T64567 CP15VC 155553400 Ki = 31.2 nM T64567 CYS29E 155553445 Ki = 860 nM T64567 C0ZO5S 155553496 IC50 = 100.9 nM T64567 C1QJ3H 155553542 Ki = 36 nM T64567 C82WXR 155553544 Ki = 28.4 nM T64567 CQM27S 155553591 Ki = 58.8 nM T64567 CQ1PE4 155553611 Ki = 31000 nM T64567 C02LSY 155553787 Ki = 220.8 nM T64567 C8SO9P 155554095 Ki = 1.6 nM T64567 C6IMR3 155554140 Ki = 0.72 nM T64567 CMEP40 155554179 Ki = 11.1 nM T64567 CE57CO 155554263 Ki = 2800 nM T64567 C0U8CG 155554286 Ki = 38.8 nM T64567 C6D9BJ 155554303 Ki = 171.1 nM T64567 C3W6RT 155554309 Ki > 50000 nM T64567 CNX5L2 155554533 Ki = 44 nM T64567 C5VLU4 155554670 Ki = 760.3 nM T64567 CM4I0O 155554763 Ki = 5400 nM T64567 CW5F4A 155554840 Ki = 19 nM T64567 CA78FQ 155555070 Ki = 260 nM T64567 C9W1ET 155555489 Ki = 235.1 nM T64567 CJ06PN 155555584 Ki > 50000 nM T64567 CV2NZ0 155555718 Ki = 35.6 nM T64567 CUY2C6 155555751 Ki = 0.36 nM T64567 CA7UK2 155555803 Ki = 111.4 nM T64567 CXNZ49 155555817 Ki = 0.24 nM T64567 CX4P1W 155555874 Ki = 24.6 nM T64567 CWB82E 155555878 Ki = 33.1 nM T64567 CKIR52 155556062 Ki = 3.9 nM T64567 C9I0QN 155556147 Ki = 17.6 nM T64567 C84MNE 155556163 Ki = 3.9 nM T64567 C5PZF2 155556257 Ki = 27.7 nM T64567 CM60WT 155556386 Ki = 45.4 nM T64567 CD4K6H 155556521 Ki = 4.7 nM T64567 CVR2X5 155556659 Ki > 100000 nM T64567 CGZ58Y 155556761 Ki = 134.8 nM T64567 C2Q3UO 155556889 Ki = 24.9 nM T64567 CYZ3K0 155556908 Ki = 73.2 nM T64567 CG8L0O 155557058 Ki = 197.9 nM T64567 CHKA19 155557282 Ki = 50.8 nM T64567 CJF9O7 155557300 Ki = 60000 nM T64567 C87GRH 155557329 Ki = 733.6 nM T64567 CRK5I0 155557428 Ki = 64.3 nM T64567 C1RMC6 155557757 Ki = 12.5 nM T64567 CNX9J2 155557875 Ki = 25.9 nM T64567 CM6NU0 155557925 Ki = 8.2 nM T64567 CWK35T 155557969 Ki = 8.3 nM T64567 CQI5Z4 155558076 Ki = 65.4 nM T64567 CK8GH2 155558119 Ki = 0.44 nM T64567 CME2Z4 155558216 Ki = 5.1 nM T64567 C70WSB 155558230 Ki = 258.2 nM T64567 CQ2ML6 155558561 Ki = 395 nM T64567 CK1RO0 155558641 Ki = 0.13 nM T64567 CH1Z2S 155558695 Ki = 58700 nM T64567 C4V2PS 155558747 Ki = 15.8 nM T64567 C6QXP8 155558748 Ki = 220 nM T64567 CZ7C0S 155558990 Ki = 2428.2 nM T64567 CI2XS3 155559081 Ki = 5.8 nM T64567 CGQ7S0 155559325 Ki = 1.4 nM T64567 C6CY3G 155559512 Ki = 0.67 nM T64567 CNT0F5 155559682 Ki = 7.5 nM T64567 CK7H8I 155559761 Ki = 13.1 nM T64567 C3Y7WJ 155560101 Ki = 9400 nM T64567 CZ2A7O 155560148 Ki = 12.1 nM T64567 CB2X0V 155560428 Ki = 12.8 nM T64567 CB5S8V 155560635 Ki = 23.5 nM T64567 COC45S 155560702 Ki = 43 nM T64567 CY1TF7 155560798 Ki = 0.56 nM T64567 C0U1NP 155560951 Ki = 34.1 nM T64567 CFY9A2 155561027 Ki = 179 nM T64567 CP3H0R 155561119 Ki = 39600 nM T64567 C3FG8W 155561198 Ki = 840 nM T64567 CSK5X2 155561354 Ki = 236.7 nM T64567 C2SZM0 155561361 Ki = 29.9 nM T64567 CHA8R0 155561556 Ki = 17.6 nM T64567 CAP5I4 155561568 Ki = 29.3 nM T64567 CU03LF 155561751 Ki = 3198.6 nM T64567 CY9N4P 155561775 Ki = 86.2 nM T64567 CU1JV7 155561839 Ki = 3066.1 nM T64567 CJ5Y6X 155561851 Ki = 211.8 nM T64567 CXE2R9 155561928 Ki = 40.7 nM T64567 C5W7MQ 155562360 Ki = 8.4 nM T64567 CG43PS 155562766 Ki = 343 nM T64567 C2FW8S 155562815 Ki = 10.1 nM T64567 CJ74ND 155563017 Ki = 35.9 nM T64567 C1J3UH 155563153 Ki = 41900 nM T64567 C7A8EX 155563186 Ki = 41.2 nM T64567 C9SH6R 155563203 Ki = 5500 nM T64567 C89MTB 155563810 Ki = 11.3 nM T64567 C0GU6P 155563888 Ki = 60.5 nM T64567 CQ40DU 155563908 Ki = 158 nM T64567 C2XB6V 155564028 Ki = 1068 nM T64567 CF7XH2 155564101 Ki = 32.3 nM T64567 CGY32K 155564210 Ki = 34.7 nM T64567 CY9M4F 155564463 Ki = 1920 nM T64567 C97TMY 155564559 Ki = 4150 nM T64567 C1K0LR 155564617 Ki = 31.7 nM T64567 CY9IW2 155564942 Ki = 2.1 nM T64567 CNV35X 155565135 Ki = 8.9 nM T64567 C0XO6Z 155565139 Ki = 90.2 nM T64567 C5XV7O 155565283 Ki = 132 nM T64567 CNL8B7 155565372 Ki = 102.4 nM T64567 CI5MV1 155565395 Ki = 54.5 nM T64567 CJ7I6Z 155565419 Ki = 19.7 nM T64567 CDF5E6 155565628 Ki = 12.6 nM T64567 C0COK6 155565635 Ki = 85 nM T64567 CT9Z5H 155565773 Ki > 50000 nM T64567 CW3N9Z 155566095 Ki = 955.3 nM T64567 COA9F8 155566222 Ki > 100000 nM T64567 CCW3L7 155566305 Ki = 665 nM T64567 C5QAM3 155566668 Ki = 13.1 nM T64567 CBV30Y 155566701 Ki = 63.2 nM T64567 CA63FB 155566994 Ki = 19.6 nM T64567 CK80EL 155567119 Ki = 61.2 nM T64567 C4TZ8Q 155567475 Ki = 14.6 nM T64567 CK0M8P 155567487 Ki = 28.6 nM T64567 CL1N9Y 155567612 Ki > 100000 nM T64567 C1MHV5 155567738 Ki = 1479 nM T64567 C29EYS 155567759 Ki = 160 nM T64567 CJ2YC4 155567804 Ki = 0.089 nM T64567 C9DOG1 155567981 Ki = 3188.1 nM T64567 CZP30I 155567991 Ki = 1465 nM T64567 CCX06Y 155568045 Ki = 74.3 nM T64567 CN5OF0 155568108 Ki > 50000 nM T64567 C2ZRJ3 155568270 Ki = 8.7 nM T64567 CG82MB 155568274 Ki = 3055.3 nM T64567 CDB8T4 155568445 Ki = 3.1 nM T64567 C52NQU 155568453 Ki = 1.9 nM T64567 C35XQY 155568474 Ki = 250.5 nM T64567 C6KR4H 155568759 Ki = 856.7 nM T64567 CH5VU6 155568899 Ki = 228.8 nM T64567 C1C2GI 155569076 Ki = 7 nM T64567 CAUR85 155569555 Ki = 230 nM T64567 D00CIW 15295 Ki = 2210000 nM T64567 D00FGB 11414131 Ki = 290 nM T64567 D00IAE 11974340 Ki = 104 nM T64567 D00IKQ 46703766 Ki = 5.7 nM T64567 D00IUB 13019 Ki = 56000 nM T64567 D00LFX 20718630 Ki = 32 nM T64567 D00NUK 2837872 Ki = 113 nM T64567 D00RDE 44246261 Ki = 4.9 nM T64567 D00RNZ 910172 Ki = 4300 nM T64567 D00SXO 2793709 Ki = 9.6 nM T64567 D00TRF 44423683 Ki = 6700 nM T64567 D00XIB 11680415 Ki = 193 nM T64567 D00XJA 711717 Ki = 5700 nM T64567 D00YEF 148885 Ki = 7 nM T64567 D01BUB 94952 Ki = 68700 nM T64567 D01CXM 52949265 Ki = 7400 nM T64567 D01EEM 462919 Ki = 9.1 nM T64567 D01FOK 52949288 Ki = 46.7 nM T64567 D01JTI 11687831 Ki = 1495 nM T64567 D01KKU 5281894 Ki = 4850 nM T64567 D01OTW 46703932 Ki = 11.7 nM T64567 D01STY 9861037 Ki = 285 nM T64567 D01UDU 11287480 Ki = 149 nM T64567 D01UYI 5281607 Ki = 2650 nM T64567 D01XFH 11851424 Ki = 113 nM T64567 D01YHK 10932611 Ki = 136 nM T64567 D02BMV 46907399 Ki = 6.3 nM T64567 D02DBP 5054 Ki = 69700 nM T64567 D02JEZ 5281426 Ki = 24.9 nM T64567 D02KDH 11160546 Ki = 175 nM T64567 D02MAK 5705744 Ki = 8030 nM T64567 D02NQK 46703924 Ki = 7.5 nM T64567 D02QGI 273 Ki = 380 nM T64567 D03APP 4386 Ki = 50 nM T64567 D03DAM 2725651 Ki = 136 nM T64567 D03KRB 45028567 Ki = 47.3 nM T64567 D03LHJ 52946829 Ki = 56.7 nM T64567 D03NBX 637308 Ki = 810 nM T64567 D03ZMQ 323 Ki > 100 nM T64567 D04BKU 148886 Ki = 54000 nM T64567 D04CVC 4687472 Ki = 245 nM T64567 D04GDW 16098578 Ki = 1180 nM T64567 D04HRS 404195 Ki = 6.4 nM T64567 D04JIN 44405179 Ki = 9280 nM T64567 D04NSN 169682 Ki = 33 nM T64567 D04POB 8482 Ki = 135 nM T64567 D04SNH 46933593 Ki = 7.8 nM T64567 D04VSP 46703768 Ki = 300 nM T64567 D05BMD 44423684 Ki = 8800 nM T64567 D05EBZ 46703769 Ki = 7.2 nM T64567 D05ETN 46703923 Ki = 313 nM T64567 D05FNN 100606 Ki = 10.1 nM T64567 D05JAJ 45028568 Ki = 9.1 nM T64567 D05KTE 6224 Ki = 4930000 nM T64567 D05QEK 44395692 Ki = 4.6 nM T64567 D05QOR 5280460 Ki = 960 nM T64567 D05QUG 45485279 Ki = 5800 nM T64567 D05RAB 45028895 Ki = 7.1 nM T64567 D05TLB 11117301 Ki = 3.5 nM T64567 D05VUA 850202 Ki = 7800 nM T64567 D05VVC 44315786 Ki = 69.7 nM T64567 D05WQF 637540 Ki > 100000 nM T64567 D05XZM 10081162 Ki = 21 nM T64567 D06DYP 234562 Ki = 5400 nM T64567 D06GPL 44405177 Ki = 250 nM T64567 D06IOI 901953 Ki = 30.4 nM T64567 D06KTD 2490720 Ki = 547 nM T64567 D06NDR 44423687 Ki = 6900 nM T64567 D06SZG 44315523 Ki = 8.2 nM T64567 D06WZG 50925425 Ki = 70.8 nM T64567 D06XNT 4119643 Ki = 136 nM T64567 D06XVV 64048 Ki = 13700 nM T64567 D06ZMH 2812287 Ki = 14 nM T64567 D06ZOM 15569045 Ki = 38.1 nM T64567 D07CBA 44391592 Ki = 525 nM T64567 D07CQI 42546 Ki = 680 nM T64567 D07IHP 44391650 Ki = 100 nM T64567 D07LYW 11537386 Ki = 282 nM T64567 D07MQB 10903168 Ki = 34 nM T64567 D07MTM 403 Ki = 517000 nM T64567 D07PNA 11660633 Ki = 3.7 nM T64567 D07PZQ 68841 Ki = 920000 nM T64567 D07QIU 625902 Ki = 883 nM T64567 D07QJJ 289 Ki = 115000 nM T64567 D07SIA 78318 Ki = 9300 nM T64567 D07TAJ 914298 Ki = 9400 nM T64567 D07UCQ 23680200 Ki = 5100 nM T64567 D07VXX 16721024 Ki = 7100 nM T64567 D07YSQ 10385283 Ki = 12 nM T64567 D07ZXR 44391576 Ki = 32.1 nM T64567 D08AOA 11543564 Ki = 2015 nM T64567 D08JCC 46703770 Ki = 7.9 nM T64567 D08JNO 52943193 Ki = 61.2 nM T64567 D08TCV 5988 Ki > 20000 nM T64567 D09CXX 16122590 Ki = 865 nM T64567 D09JPC 16402 Ki = 410 nM T64567 D09LUD 4229592 Ki = 18 nM T64567 D09PWX 8739 Ki = 26 nM T64567 D09TKG 25044690 Ki = 12 nM T64567 D09UQM 97463 Ki = 540 nM T64567 D09USO 5277466 IC50 = 7629 nM T64567 D09WSJ 19772348 Ki = 23 nM T64567 D09WVV 8111 Ki = 10600 nM T64567 D0A0YX 5143 Ki = 100 nM T64567 D0A1CM 5281855 Ki = 9370 nM T64567 D0A4TC 446504 Ki = 7800 nM T64567 D0A6HS 6852129 Ki = 14 nM T64567 D0AU0M 637542 Ki = 5330 nM T64567 D0B4IN 375084 Ki = 653 nM T64567 D0B5GC 11349 Ki = 5540 nM T64567 D0BD0K 405487 Ki = 6 nM T64567 D0BM2T 44577440 Ki = 24 nM T64567 D0C6ED 44564283 Ki = 61.6 nM T64567 D0C7LR 313 Ki = 33000000 nM T64567 D0C7WG 135932620 Ki = 6.1 nM T64567 D0CM3O 446142 Ki = 31300000 nM T64567 D0D0BO 180598 Ki = 181 nM T64567 D0D4OV 20043772 Ki = 4 nM T64567 D0D6UR 12394434 Ki = 6200 nM T64567 D0DY9U 23645365 Ki = 65 nM T64567 D0E0RW 69894 Ki = 7370 nM T64567 D0E8CC 18794 Ki = 42 nM T64567 D0EH0S 52943164 Ki = 58.2 nM T64567 D0EJ9B 66827 Ki > 50000 nM T64567 D0EY2F 52949920 Ki = 8015 nM T64567 D0F3UR 690836 Ki = 23.7 nM T64567 D0F7KC 14116752 Ki = 78.3 nM T64567 D0F7SO 94464 Ki = 32 nM T64567 D0FU0K 23354226 Ki = 7.7 nM T64567 D0G0BJ 51000408 Ki > 50000 nM T64567 D0G0FJ 11206245 Ki = 48 nM T64567 D0G0OP 44423685 Ki = 9200 nM T64567 D0G0ZI 403788 Ki > 50000 nM T64567 D0G3BI 25090 Ki = 48 nM T64567 D0G6OW 23675285 Ki = 770000 nM T64567 D0G9NE 11659798 Ki = 108 nM T64567 D0H3NS 10752 Ki = 6500 nM T64567 D0H4CF 44246267 Ki = 5.9 nM T64567 D0HN0R 11623958 Ki = 30 nM T64567 D0I5YQ 44405178 Ki = 2420 nM T64567 D0IU3X 44405186 Ki = 7730 nM T64567 D0J1PZ 2723687 Ki = 9500 nM T64567 D0J2AE 7377 Ki = 238 nM T64567 D0J3SP 11718391 Ki = 33 nM T64567 D0J7GU 46703929 Ki = 47 nM T64567 D0J7KJ 52940758 Ki = 7580 nM T64567 D0K1FG 5411574 Ki = 73 nM T64567 D0K3LN 3510137 Ki = 83 nM T64567 D0KB6T 721954 Ki = 73 nM T64567 D0KZ2D 11638641 Ki = 37.5 nM T64567 D0L2GD 60167587 Ki = 4770000 nM T64567 D0L4FM 11030308 Ki = 63 nM T64567 D0L5TZ 20195365 Ki = 8400 nM T64567 D0L5XK 92249 Ki = 7640 nM T64567 D0LJ5P 44457221 Ki = 8.1 nM T64567 D0LU4S 156219 Ki = 4900 nM T64567 D0M3PO 69561 Ki = 24 nM T64567 D0M5MI 4306515 IC50 > 100000 nM T64567 D0M6RM 7365 Ki = 55000 nM T64567 D0M9IQ 23665438 Ki = 5850 nM T64567 D0N1AW 45485270 Ki = 8400 nM T64567 D0N5KX 44391625 Ki = 61.6 nM T64567 D0N8LR 847760 Ki = 106 nM T64567 D0N8VZ 11583423 Ki = 250 nM T64567 D0NN3Q 78105 Ki = 265 nM T64567 D0NS0E 220188 Ki = 480 nM T64567 D0O0UE 729977 Ki = 84 nM T64567 D0O4KL 11640067 Ki = 3.2 nM T64567 D0O6ZD 14101447 Ki = 72.3 nM T64567 D0O8WV 11536481 Ki = 2320 nM T64567 D0OC4B 5357479 Ki = 47.2 nM T64567 D0OI1H 72894 Ki = 33 nM T64567 D0OT5L 1631814 Ki = 8100 nM T64567 D0P6AM 3526523 Ki = 269 nM T64567 D0Q0EK 318174 Ki = 175 nM T64567 D0Q0XO 4258082 Ki = 79 nM T64567 D0Q1EI 3084733 Ki = 68 nM T64567 D0Q2XB 75928 Ki = 944 nM T64567 D0Q5VB 46704078 Ki = 15.8 nM T64567 D0Q7DJ 10742 Ki = 8200 nM T64567 D0R4KQ 46704077 Ki = 7.8 nM T64567 D0R7QY 127676 Ki = 30 nM T64567 D0RB0D 44268050 Ki = 4100 nM T64567 D0RK7J 235259 Ki = 112 nM T64567 D0S0RK 10680 Ki = 4130 nM T64567 D0S2II 308405 Ki = 454 nM T64567 D0S3RZ 9954405 Ki = 58 nM T64567 D0SF3B 11529486 Ki = 3.4 nM T64567 D0T2YZ 3253857 Ki = 139 nM T64567 D0T3NP 7456 Ki = 5500 nM T64567 D0T9BB 52950111 Ki = 37.8 nM T64567 D0TY8X 31036 Ki = 16 nM T64567 D0U4BB 10748 Ki = 9800 nM T64567 D0UM1I 12554666 Ki = 4.9 nM T64567 D0UN0E 12195854 Ki = 8500 nM T64567 D0V0FY 52946831 Ki = 50.2 nM T64567 D0V5OW 46907400 Ki = 11.8 nM T64567 D0V9EN 689043 Ki = 7870 nM T64567 D0VD7H 84724 Ki = 41 nM T64567 D0W1AW 4234241 Ki = 643 nM T64567 D0W1OR 7424 Ki = 4410 nM T64567 D0W9VC 670143 Ki = 19 nM T64567 D0X0PO 20043771 Ki = 13.2 nM T64567 D0X1MY 2723847 Ki = 9300 nM T64567 D0X5HL 15107 Ki = 510 nM T64567 D0X6IE 4422372 Ki = 31 nM T64567 D0X9LJ 788811 Ki = 290 nM T64567 D0Y1XM 44423686 Ki = 7600 nM T64567 D0Y3TZ 370 Ki = 6990 nM T64567 D0YD9F 822774 Ki = 52 nM T64567 D0YU8J 1502014 Ki = 264 nM T64567 D0YZ5G 5281416 Ki = 36.4 nM T64567 D0Z1HY 67136 Ki = 39 nM T64567 D0Z6TM 3558590 Ki = 105 nM T64567 D0ZC3W 6269 Ki = 460 nM T49542 D0E3TC 44259 IC50 = 261 nM T49542 C3VRO9 44557921 IC50 > 10000 nM T49542 C86YRV 58688296 IC50 > 30000 nM T49542 C8AT5N 58688313 IC50 > 30000 nM T49542 C09YWX 58688317 IC50 > 12500 nM T49542 C4Q2HL 58688342 IC50 = 11910 nM T49542 C0LK4S 58688380 IC50 > 30000 nM T49542 CNVK41 58688409 IC50 > 30000 nM T49542 CJI0Q4 58688436 IC50 > 30000 nM T49542 CK1AO4 58688444 IC50 > 30000 nM T49542 CZ0J6F 58688467 IC50 > 30000 nM T49542 CPE98M 58688474 IC50 > 30000 nM T49542 CDOK25 58688484 IC50 > 30000 nM T49542 CHO5G0 58688561 IC50 > 30000 nM T49542 CP2JK1 58688569 IC50 > 30000 nM T49542 CIV53P 58688575 IC50 = 1133 nM T49542 C2T8UL 58688642 IC50 > 30000 nM T49542 CV63UL 67240318 IC50 > 10000 nM T49542 CIJ5L9 70682556 IC50 > 30000 nM T49542 C9IB8C 70684645 IC50 = 2265 nM T49542 CH08ZN 70690951 IC50 > 30000 nM T49542 CK0CH3 70697188 IC50 > 30000 nM T49542 C3B4HT 136003186 IC50 > 30000 nM T49542 D0F6NZ 58688690 IC50 = 2198 nM T49542 D0FC4Y 46192505 IC50 = 455 nM T49542 D0S0XD 58688563 IC50 > 30000 nM T60526 D02AUB 9811353 IC50 > 500000 nM T60526 C1GDY7 587790 IC50 = 38500 nM T60526 C96KNY 643990 IC50 > 1000000 nM T60526 CZ98HT 9977686 IC50 > 500000 nM T60526 C4Z0FP 11258464 IC50 = 13600 nM T60526 C62DAO 16114614 IC50 = 1400 nM T60526 C1ET3V 16114615 IC50 > 500000 nM T60526 CQ90BS 16114616 IC50 = 3100 nM T60526 CA4MJ7 16114618 IC50 = 30800 nM T60526 CWGO19 16114619 IC50 = 4200 nM T60526 CTC76N 16114620 IC50 = 109000 nM T60526 CM7Z2R 16115893 IC50 = 1500 nM T60526 C41WNZ 16116039 IC50 = 8700 nM T60526 CUE4D8 16116040 IC50 = 64900 nM T60526 C2EHS8 16116042 IC50 = 46600 nM T60526 CTG1J6 16116159 IC50 = 2300 nM T60526 CZH0G1 16116162 IC50 = 26200 nM T60526 C5GZB3 16116163 IC50 = 64500 nM T60526 CG05BP 16116164 IC50 > 500000 nM T60526 CKI2E4 16116165 IC50 = 105100 nM T60526 C5Q4GR 16116166 IC50 = 85800 nM T60526 C7F1DY 16116286 IC50 = 21300 nM T60526 CU4OF0 16116421 IC50 = 154400 nM T60526 C89WXF 16116422 IC50 = 14600 nM T60526 C82KGR 16116555 IC50 = 41700 nM T60526 C9DME7 16116556 IC50 = 4300 nM T60526 CU2IB8 16116557 IC50 = 9800 nM T60526 CTXB17 16116558 IC50 = 37600 nM T60526 CFU0D9 16116559 IC50 = 244000 nM T60526 C7WJ0Y 16725848 IC50 = 790 nM T60526 CC12EZ 23709469 IC50 = 30000 nM T60526 CQP9G7 44304820 IC50 > 1000000 nM T60526 CD1Y6W 44340382 IC50 = 114000 nM T60526 CC7G9J 44340394 IC50 = 170000 nM T60526 C2Q7LW 44340567 IC50 = 3000 nM T60526 CZG4T2 44340638 IC50 = 11000 nM T60526 CK1GA0 44340639 IC50 = 1000 nM T60526 CICW90 44356343 IC50 = 12000 nM T60526 C1VH5G 44356439 IC50 = 3800 nM T60526 CK7WE9 44356515 IC50 > 500000 nM T60526 CPM04F 44356616 IC50 = 2400 nM T60526 C8CR4F 44356617 IC50 = 200000 nM T60526 CXL0S8 44387278 IC50 > 1000000 nM T60526 CIAL79 44387290 IC50 = 35000 nM T60526 CHIF62 44387291 IC50 = 420000 nM T60526 C6FK5A 44387293 IC50 = 220000 nM T60526 C7WPK9 44387294 IC50 > 1000000 nM T60526 CPQ09T 44387295 IC50 > 1000000 nM T60526 CPT5K3 44387297 IC50 > 1000000 nM T60526 C0ZIP8 44420653 IC50 = 3300 nM T60526 C5QXG3 44420654 IC50 = 5700 nM T60526 C2S9CH 44420657 IC50 = 1600 nM T60526 C8Y1HG 44420659 IC50 = 1600 nM T60526 CQ08EK 44420661 IC50 = 1100 nM T60526 CA9T5O 44420662 IC50 = 9700 nM T60526 CEPH60 71452644 IC50 = 35000 nM T60526 CN0ZI6 71458017 IC50 = 106000 nM T60526 CGE8R2 71715994 IC50 = 3100 nM T60526 C0FR3U 71716010 IC50 = 4000 nM T60526 C3S7VA 71716029 IC50 = 3000000 nM T60526 C3JQ6N 71716030 IC50 = 560000 nM T60526 CEO6H7 71716031 IC50 = 1400000 nM T60526 C6C0ZR 71716033 IC50 = 3000000 nM T60526 CS7T0Y 71717230 IC50 = 5000000 nM T60526 CK27AE 71717234 IC50 = 750000 nM T60526 C8P0KB 71717843 IC50 = 4100000 nM T60526 CLN8X2 71717844 IC50 = 3000000 nM T60526 CCO93Y 71719057 IC50 = 40000 nM T60526 CH42FQ 71719059 IC50 = 600000 nM T60526 CI6Z9O 71719670 IC50 = 1000000 nM T60526 CQR6H7 71719671 IC50 = 750000 nM T60526 C2XBN3 71719672 IC50 = 300000 nM T60526 C32CAX 71720271 IC50 = 2000000 nM T60526 C3Y5QT 71720273 IC50 = 500000 nM T60526 C8TE5P 76335199 IC50 = 30000 nM T60526 CO2DA9 90664124 IC50 > 1000000 nM T60526 CKZP37 90664125 IC50 > 1000000 nM T60526 CJ3O0E 90664264 IC50 = 4000 nM T60526 C6KN7R 90664265 IC50 = 2340 nM T60526 C15YGB 118719302 IC50 = 1800 nM T60526 CI3VJ0 118719304 IC50 = 1600 nM T60526 CZH6T3 118719305 IC50 = 700 nM T60526 C4BGF1 118719306 IC50 = 800 nM T60526 D0E9NT 11874 IC50 = 15200 nM T60526 D0Y3TZ 370 IC50 = 27600 nM T57006 D0E3TC 44259 IC50 = 56.3 nM T57006 C2ICS7 25065806 IC50 > 1000 nM T57006 CV63UL 67240318 IC50 > 10000 nM T57006 CQ2OB9 90292687 IC50 = 665 nM T57006 C9WGB8 127035904 IC50 = 2500 nM T57006 CXC69T 137321158 IC50 = 190 nM T57006 C2MD1Q 155513187 IC50 > 10000 nM T57006 D02BXJ 46864270 IC50 = 4.2 nM T57006 D05FXD 44478401 IC50 = 1118 nM T57006 D0X8BU 71718651 IC50 = 2100 nM T47623 D04KNL 57412324 Ki = 6.1 nM T47623 C5V3DJ 1048811 IC50 = 10000 nM T47623 CJAQ62 1104017 IC50 = 1200 nM T47623 C2GNV1 1271221 IC50 = 8000 nM T47623 CPV8F2 2236365 IC50 = 4000 nM T47623 CYIN23 2797588 IC50 = 300000 nM T47623 C4ZQ3P 3091496 IC50 = 1500 nM T47623 C59FTW 9828828 IC50 = 398.11 nM T47623 CL4S7G 9913234 IC50 = 199.53 nM T47623 CKE6J9 9961858 IC50 = 8000 nM T47623 CJWH38 9988952 IC50 = 2000 nM T47623 CH7QO6 10030498 IC50 = 200 nM T47623 C2IUD6 10074971 IC50 = 1000 nM T47623 C9SIX7 10098264 IC50 = 1500 nM T47623 C14CAF 10196332 IC50 = 500 nM T47623 C9J5TI 10232463 IC50 = 5000 nM T47623 C8L3YS 10256575 IC50 = 300 nM T47623 C27EDN 10316085 IC50 = 25000 nM T47623 CD1J0O 10412145 IC50 = 450 nM T47623 CXY51U 10436279 IC50 = 3467.37 nM T47623 CO3RA4 10480716 IC50 = 3000 nM T47623 CWRO82 11014442 IC50 > 100000 nM T47623 CE89AN 11179557 IC50 = 75 nM T47623 CVU39C 11293715 IC50 = 270 nM T47623 CY2DR4 11305158 IC50 = 930 nM T47623 CV2U3R 11364514 IC50 = 370 nM T47623 CB05RT 11513613 IC50 = 250 nM T47623 CN0D2Q 11563127 IC50 = 350 nM T47623 CDB9F2 11663697 IC50 = 290 nM T47623 CSP8Q7 11705939 IC50 = 199.53 nM T47623 CG3P8W 11712551 IC50 = 150 nM T47623 CN43BG 14217343 IC50 = 12000 nM T47623 C9IU0C 15999192 IC50 > 15000 nM T47623 C3JQ4E 16439879 IC50 = 1000 nM T47623 CJN3T0 21120908 IC50 = 1000 nM T47623 C3U2QM 21884300 IC50 = 4466.84 nM T47623 CPD4C1 21884333 IC50 > 10000 nM T47623 CM27ZC 21884347 IC50 = 3000 nM T47623 C5OFU6 21884358 IC50 = 3019.95 nM T47623 CB80LT 21884371 IC50 = 600 nM T47623 C1DQ5T 21884395 IC50 = 900 nM T47623 CL7OW9 21884416 IC50 = 398.11 nM T47623 C7JCL2 21884458 IC50 = 3000 nM T47623 CRY7D9 21884463 IC50 = 398.11 nM T47623 C8HL5I 21884468 IC50 = 1995.26 nM T47623 CQ86BP 21884541 IC50 = 3000 nM T47623 CO05GB 21884542 IC50 = 2500 nM T47623 C9Y1RV 21884564 IC50 = 1500 nM T47623 CA6Y3O 21884578 IC50 = 3981.07 nM T47623 CDJE25 21884589 IC50 = 1000 nM T47623 CQ50YM 21884595 IC50 = 1288.25 nM T47623 CLF8C9 21884600 IC50 = 250 nM T47623 CFAC14 21884606 IC50 = 5000 nM T47623 C24YVK 21884635 IC50 = 800 nM T47623 C9ZUL2 27844286 IC50 > 15000 nM T47623 C92HQT 44339670 IC50 = 3000 nM T47623 C8L2MT 44339681 IC50 = 199.53 nM T47623 CZIJ69 44339689 IC50 = 400 nM T47623 C0SU1N 44339698 IC50 = 750 nM T47623 C34XGM 44339701 IC50 = 2000 nM T47623 CI23OV 44339702 IC50 = 2000 nM T47623 C4ZX8J 44339703 IC50 = 800 nM T47623 CRLW68 44339721 IC50 = 8912.51 nM T47623 C9DZA2 44339754 IC50 = 600 nM T47623 C1C3MD 44339760 IC50 = 2500 nM T47623 C5MZ8U 44339774 IC50 = 398.11 nM T47623 C76EWZ 44339782 IC50 = 1000 nM T47623 CF78RM 44339823 IC50 = 500 nM T47623 CVW0A2 44339856 IC50 = 602.56 nM T47623 C9OIH1 44339881 IC50 > 10000 nM T47623 C65HEG 44339891 IC50 = 2500 nM T47623 CTQ0Z7 44339892 IC50 = 200 nM T47623 C2I4JL 44339893 IC50 = 3000 nM T47623 C1SIL0 44339897 IC50 > 10000 nM T47623 CBI1D6 44339955 IC50 > 10000 nM T47623 CY6R3F 44340019 IC50 = 8912.51 nM T47623 CQ8C9H 44340022 IC50 = 446.68 nM T47623 C8GQP1 44340027 IC50 = 3000 nM T47623 C1R7CG 44340037 IC50 > 10000 nM T47623 CTD76W 44340051 IC50 > 10000 nM T47623 CF7EO8 44402002 IC50 = 600 nM T47623 CN4K0E 44402023 IC50 > 10000 nM T47623 C0JT7Q 44402024 IC50 = 350 nM T47623 CHD62Z 44402162 IC50 = 8500 nM T47623 C4XSW3 44402163 IC50 = 2500 nM T47623 C7P4MF 44402193 IC50 = 400 nM T47623 CL75RX 44402209 IC50 = 3000 nM T47623 CUM28T 44402210 IC50 = 800 nM T47623 CY3FJ1 44402233 IC50 = 398.11 nM T47623 C61YMT 44402336 IC50 = 450 nM T47623 C9IU4W 44402337 IC50 = 2500 nM T47623 CWFV78 44402338 IC50 = 1995.26 nM T47623 C9TAW0 44402342 IC50 = 794.33 nM T47623 C2IZ5P 44402362 IC50 = 8500 nM T47623 CSR5U7 44402363 IC50 > 10000 nM T47623 CDZH89 44402366 IC50 > 10000 nM T47623 C2W6SU 44402379 IC50 > 30000 nM T47623 C7OKP4 44402380 IC50 = 8000 nM T47623 CC08ZE 44402381 IC50 = 398.11 nM T47623 C8QBK7 44402399 IC50 = 3000 nM T47623 CQM8O5 44402400 IC50 = 4000 nM T47623 C0KG6Q 44402407 IC50 = 398.11 nM T47623 CZFA72 44402408 IC50 = 691.83 nM T47623 CP3ZX0 44402409 IC50 = 3019.95 nM T47623 C9LD0E 44402422 IC50 = 501.19 nM T47623 C4E5HS 44402423 IC50 = 741.31 nM T47623 CUR82F 44402425 IC50 > 30000 nM T47623 CQ8N5Z 44402443 IC50 = 2500 nM T47623 C6A2GW 44402444 IC50 = 3000 nM T47623 CJ58BX 44402473 IC50 = 350 nM T47623 CSG43T 44402474 IC50 = 741.31 nM T47623 CL2I4X 44402494 IC50 = 3467.37 nM T47623 CI7QR9 44402495 IC50 = 420 nM T47623 C1GC8U 44402501 IC50 = 3000 nM T47623 C4NUA0 44402523 IC50 = 398.11 nM T47623 CN96MK 44402524 IC50 = 3000 nM T47623 CI90LV 44402539 IC50 = 300 nM T47623 CHJ1T5 44402540 IC50 = 3000 nM T47623 CHI84R 44402541 IC50 = 3019.95 nM T47623 CA3UK6 44402554 IC50 = 1500 nM T47623 C52ZXY 44402556 IC50 = 741.31 nM T47623 C29ZBF 44402558 IC50 = 3981.07 nM T47623 CQIT23 44402573 IC50 = 794.33 nM T47623 C5H9KC 44402574 IC50 = 2500 nM T47623 CIO54X 44402575 IC50 = 2500 nM T47623 CXR34U 44402576 IC50 = 300 nM T47623 C3X4PO 44402592 IC50 = 300 nM T47623 CVC5X1 44402608 IC50 = 5495.41 nM T47623 C8TFA9 44402609 IC50 = 691.83 nM T47623 CC6GL9 44402641 IC50 = 199.53 nM T47623 CVM0J9 44402643 IC50 = 2500 nM T47623 COW8J9 44402644 IC50 = 750 nM T47623 CPHK80 44402665 IC50 = 2511.89 nM T47623 CW1V8Z 44402666 IC50 = 3000 nM T47623 C9JSY4 44405111 IC50 = 2020 nM T47623 CA2O7I 44405114 IC50 = 1850 nM T47623 CG1W5E 44405116 IC50 = 1830 nM T47623 C0C5GE 44405117 IC50 = 1640 nM T47623 CC6RO5 44406239 IC50 = 2200 nM T47623 CS69DO 44406240 IC50 = 11000 nM T47623 C27XGJ 44406329 IC50 = 2300 nM T47623 C59QJB 44406357 IC50 = 5700 nM T47623 C9KP0A 44406363 IC50 = 6100 nM T47623 C94EMV 44406369 IC50 = 1150 nM T47623 C5VLR4 44406371 IC50 = 1600 nM T47623 CUDF57 44406378 IC50 = 930 nM T47623 C9RA4H 44406400 IC50 = 1300 nM T47623 C4ARO1 44406404 IC50 = 1100 nM T47623 C5A2LN 44406405 IC50 = 2700 nM T47623 CZ67NL 44406410 IC50 > 15000 nM T47623 C4MK8T 44406412 IC50 = 150 nM T47623 C31WEG 44406422 IC50 = 150 nM T47623 CDZ9V3 44406440 IC50 > 15000 nM T47623 CTKX15 44406445 IC50 > 15000 nM T47623 C82FLG 44406461 IC50 = 1000 nM T47623 CFLR58 44406473 IC50 > 15000 nM T47623 CK04SQ 44406474 IC50 > 15000 nM T47623 CG3RI5 44406485 IC50 = 3420 nM T47623 C2VG7Q 44406515 IC50 = 910 nM T47623 CCY34F 44406530 IC50 = 870 nM T47623 CF15YS 44406531 IC50 = 900 nM T47623 CGW6E1 44450830 IC50 = 4150 nM T47623 CTPM18 44450876 Ki = 240 nM T47623 CP7UK2 44450934 Ki = 280 nM T47623 C95KRJ 44450956 Ki = 200 nM T47623 CPT2F6 44451051 IC50 = 1570 nM T47623 CKG7W6 44576544 IC50 = 346.74 nM T47623 CT2V5H 44576545 IC50 = 346.74 nM T47623 C60QPT 44576546 IC50 = 794.33 nM T47623 CE28HC 44576550 IC50 = 2511.89 nM T47623 C04WOV 44576551 IC50 = 3019.95 nM T47623 C5NTK0 44576552 IC50 = 1995.26 nM T47623 C5D0PY 44576553 IC50 = 1995.26 nM T47623 C93KNB 44576554 IC50 = 794.33 nM T47623 CQW7O6 44585480 IC50 = 3019.95 nM T47623 CJ23LT 44585486 IC50 = 446.68 nM T47623 CA3RX8 53319770 IC50 = 2690 nM T47623 C6QU4Y 53321097 Ki = 7.9 nM T47623 CNW03R 57412318 Ki = 5.8 nM T47623 C70KOE 57412320 Ki = 6 nM T47623 CC2T0R 57412326 Ki = 3.7 nM T47623 CV2NT7 57412411 Ki = 22.3 nM T47623 CS7Z0B 57412413 Ki = 6.4 nM T47623 C53ZQN 57412415 Ki = 20 nM T47623 C37HLI 57412417 Ki = 9.1 nM T47623 C1YAG5 57412494 Ki = 8.5 nM T47623 CLT3V1 57412578 Ki = 10.5 nM T47623 CVW0L9 57412675 Ki = 8.4 nM T47623 CFAQ01 57412842 Ki = 16 nM T47623 CL09RE 57412932 Ki = 9.1 nM T47623 CKU9X6 57412934 Ki = 11.3 nM T47623 CGWR86 57413121 Ki = 111 nM T47623 C6B1AJ 57413208 Ki = 30 nM T47623 CQ2U9T 70696809 Ki = 5.5 nM T47623 C03JGD 71716558 IC50 = 26000 nM T47623 C5DO9E 71718394 IC50 > 100000 nM T47623 CC7F0J 71720833 IC50 = 24000 nM T47623 C1NIX9 71720834 IC50 = 200 nM T47623 CRZ62F 73355036 IC50 = 26600 nM T47623 CWV85J 90643920 IC50 = 66390 ug.mL-1 T47623 CS9YW5 90664063 IC50 = 10000 nM T47623 CNI8G2 90664064 IC50 = 10000 nM T47623 CO87ET 135341056 IC50 > 10000 nM T47623 C1KY4J 135341058 IC50 > 10000 nM T47623 C2PZM4 135341060 IC50 = 820 nM T47623 C42TWV 135341064 IC50 > 10000 nM T47623 CVGN27 135341067 IC50 = 1330 nM T47623 C3W1HY 135341069 IC50 = 2560 nM T47623 C0VR5G 135341073 IC50 = 5700 nM T47623 CRN7G3 135341075 IC50 = 2290 nM T47623 C6LI4G 135341076 IC50 = 640 nM T47623 CHG80Q 135341078 IC50 = 1590 nM T47623 CE8LZ6 135341080 IC50 = 3460 nM T47623 CAQ1D6 135341083 IC50 = 2860 nM T47623 CG84VL 135341091 IC50 = 980 nM T47623 CIX29Z 135341094 IC50 = 990 nM T47623 CQG0Z5 135341095 IC50 = 1810 nM T47623 C0P9IE 135341096 IC50 = 1400 nM T47623 CW6Q4S 135341098 IC50 > 10000 nM T47623 CU5IO2 135341099 IC50 = 180 nM T47623 CDS0I4 135341105 IC50 = 3200 nM T47623 C8GDC3 135341108 IC50 > 10000 nM T47623 C12SIM 139667025 IC50 = 1190 nM T47623 C8A6HG 139667030 IC50 > 10000 nM T47623 C9B1QA 142438522 IC50 > 10000 nM T47623 CK8NL3 142438524 IC50 = 6020 nM T47623 CLY67W 142438526 IC50 = 80 nM T47623 C2SB8O 142438535 IC50 = 160 nM T47623 CN2M3F 145964854 IC50 = 5640 nM T47623 C7LRJ4 145966441 IC50 = 1720 nM T47623 CP1U9S 145967352 IC50 = 8530 nM T47623 CBPZ42 145969165 IC50 = 860 nM T47623 C19YCV 145973251 IC50 = 1480 nM T47623 C7HEZ1 145976385 IC50 = 3400 nM T47623 CU59WS 145977077 IC50 = 660 nM T47623 CR7E0B 145978983 IC50 = 720 nM T47623 CL03NS 145979718 IC50 = 2730 nM T47623 C56JRE 145980047 IC50 = 9170 nM T47623 CBF0N7 145980201 IC50 = 1760 nM T47623 CS9M0U 145980244 IC50 = 450 nM T47623 CA4SY5 145980482 IC50 > 10000 nM T47623 CEXM96 145981430 IC50 > 10000 nM T47623 CRX8G9 145982170 IC50 = 5 nM T47623 C5OAL0 145982269 IC50 > 10000 nM T47623 C1K8XV 145983015 IC50 = 16000 nM T47623 CX4SM2 145986393 IC50 = 4870 nM T47623 C1WNC9 145987521 IC50 = 820 nM T47623 C0DRG2 145987682 IC50 > 10000 nM T47623 CB8R9H 145988144 IC50 > 10000 nM T47623 CAV30Y 145988229 IC50 = 370 nM T47623 C0ECJ1 145988870 IC50 > 10000 nM T47623 CV9H2T 145989060 IC50 > 10000 nM T47623 C8L3RE 145989439 IC50 > 10000 nM T47623 CSY19L 145990214 IC50 > 10000 nM T47623 C96IFJ 145990605 IC50 = 2610 nM T47623 C9TE1A 145993329 IC50 > 10000 nM T47623 CQ05FA 145994103 IC50 > 10000 nM T47623 CKWP81 155513270 IC50 = 9961 nM T47623 C9T4OW 155519605 IC50 = 8225 nM T47623 C7WJ8D 155529062 IC50 = 3012 nM T47623 C06YTD 155529183 IC50 = 42060 nM T47623 CB7YC0 155532019 IC50 = 9537 nM T47623 CJR63Y 155533734 IC50 = 8118 nM T47623 CXI57M 155537182 IC50 = 11210 nM T47623 C4MDF9 155539354 IC50 = 3940 nM T47623 C1UYW3 155546936 IC50 = 10790 nM T47623 C0D5YW 155548172 IC50 = 393 nM T47623 CF3O6S 155549743 IC50 = 41680 nM T47623 C89TVD 155555142 IC50 = 12390 nM T47623 CUPI64 155557484 IC50 = 2690 nM T47623 CB6VQ5 155563498 IC50 = 11961 nM T47623 D08BSQ 54678922 IC50 = 17000 nM T99160 D04LVK 57379345 IC50 = 2240 nM T99160 D0W5HK 216239 IC50 = 262 nM T99160 D03HUX 49792852 IC50 > 10000 nM T99160 D03LWG 53235510 IC50 > 10000 nM T99160 D06EGV 44603533 IC50 = 109 nM T99160 D07EHV 44814409 IC50 > 10000 nM T99160 D07XOV 118598754 IC50 = 1 nM T99160 D0E3TC 44259 IC50 = 20.3 nM T99160 D0O6WV 24794418 IC50 > 500 nM T99160 D03BNU 59604787 IC50 > 10000 nM T99160 D0ZH4I 76071870 IC50 = 14 nM T99160 CVQ15R 459521 IC50 = 17000 nM T99160 C2Y9UB 1515243 IC50 = 12000 nM T99160 CK5WN4 1515244 IC50 = 6000 nM T99160 C15MJS 2239542 Ki > 10000 nM T99160 C8SYF6 2725997 IC50 = 20000 nM T99160 CI9N4S 2735305 IC50 = 20000 nM T99160 CJGT05 2735393 IC50 = 11000 nM T99160 C6R5VD 2735821 IC50 = 5200 nM T99160 CPI2C5 2775690 IC50 = 7100 nM T99160 CE16XS 2780715 IC50 = 36000 nM T99160 CU0V1A 4739100 IC50 = 2900 nM T99160 CVN8T9 10379252 IC50 = 720 nM T99160 CJR7W4 13521419 IC50 = 900 nM T99160 CD1I7O 14623308 IC50 = 11 nM T99160 CY8L7E 24896769 IC50 > 10000 nM T99160 CPAO21 26081407 IC50 > 10000 nM T99160 CR2W7S 28855509 Ki = 164 nM T99160 CZ63DC 39817743 IC50 = 1500 nM T99160 C5QVB8 44518236 IC50 = 580 nM T99160 CU3RF1 45139989 IC50 > 10000 nM T99160 CQGZ06 45139991 IC50 > 10000 nM T99160 CQ7W3Y 46182043 Ki = 4050 nM T99160 CQJ1W7 46182661 Ki = 68 nM T99160 C7ON5A 46233287 IC50 > 10000 nM T99160 CLS29B 46872626 IC50 > 10000 nM T99160 C08EBI 46937430 IC50 = 575 nM T99160 CRA74I 49842779 IC50 > 10000 nM T99160 CF91RS 49843531 IC50 > 10000 nM T99160 C2Y6QS 50938552 IC50 > 10000 nM T99160 C9NYP4 51036677 IC50 > 10000 nM T99160 C4WRY3 51037112 IC50 > 10000 nM T99160 CRI28Z 51037948 IC50 > 10000 nM T99160 C2W9OA 53324451 IC50 = 150 nM T99160 C5TI4A 53494955 IC50 > 10000 nM T99160 C1XS2J 54760383 IC50 = 3200 nM T99160 CV56NF 57428036 IC50 = 3600 nM T99160 CI10DA 58452049 IC50 = 184000 nM T99160 C97ZGJ 58539301 IC50 = 600 nM T99160 C08RDP 58714747 IC50 > 10000 nM T99160 C1HSE0 67035086 IC50 = 1100 nM T99160 CWI6K5 67035106 IC50 > 10000 nM T99160 CV63UL 67240318 IC50 > 10000 nM T99160 CRF2P7 68233509 Ki > 10000 nM T99160 C8I7GC 68293638 IC50 > 10000 nM T99160 CD56XK 68293660 IC50 > 10000 nM T99160 C29IXH 70683189 IC50 > 10000 nM T99160 CMX61J 70683190 IC50 > 10000 nM T99160 CRL16Z 70683191 IC50 > 10000 nM T99160 CD3Z6H 70691589 IC50 = 1610 nM T99160 CR8OG6 70691590 IC50 > 10000 nM T99160 CLT7F0 70691591 IC50 = 1350 nM T99160 CZ7S5O 70691592 IC50 > 10000 nM T99160 C8QW3C 70691593 IC50 > 10000 nM T99160 CZOW87 70691594 IC50 > 10000 nM T99160 CFQ62O 70695787 IC50 > 10000 nM T99160 CCN01X 71547862 IC50 > 10000 nM T99160 CH45ZR 71744719 IC50 = 41 nM T99160 C8YA3T 71766208 IC50 = 11 nM T99160 C5CDM4 71766212 IC50 = 454 nM T99160 C6P9HZ 71766360 IC50 = 86 nM T99160 C2PAK9 73438493 IC50 = 10 nM T99160 C4U5NV 73442760 IC50 = 760000 nM T99160 CHI51J 76070594 IC50 = 33 nM T99160 C8VAD5 76070929 IC50 = 12 nM T99160 CB4V1R 76071142 IC50 = 44 nM T99160 CBAT06 76071144 IC50 = 16 nM T99160 C7SH1T 76071506 IC50 = 8 nM T99160 CS87EI 76071624 IC50 = 32 nM T99160 CGC0K4 76071869 IC50 = 11 nM T99160 C1MY3O 86290971 IC50 = 370 nM T99160 CGD0S5 89825760 IC50 = 72 nM T99160 CR5H9I 89826764 IC50 = 336 nM T99160 C7GC8K 89826796 IC50 = 143 nM T99160 C1IA0Q 89826982 IC50 = 25 nM T99160 CMJY71 89827041 IC50 = 502 nM T99160 CT6W0Y 89835558 IC50 = 26 nM T99160 CG7YI5 90167717 IC50 = 43000 nM T99160 CY0UC4 90645194 IC50 > 10000 nM T99160 CBP5K7 91183030 IC50 = 22 nM T99160 CDM21G 117737362 IC50 = 389 nM T99160 CWL6D7 117737365 IC50 = 217 nM T99160 CR6G8P 118242667 Ki = 500 nM T99160 C01HYG 118598634 IC50 = 1.2 nM T99160 CL5W7Y 118598693 IC50 = 1.8 nM T99160 C9F0JN 118598698 IC50 = 2.3 nM T99160 C2KW9T 118598721 IC50 = 57 nM T99160 CDSW54 118598782 IC50 = 1.5 nM T99160 C2MI8L 118598816 IC50 = 0.68 nM T99160 CL0Q6D 118598855 IC50 = 1 nM T99160 C1X9MR 118598890 IC50 = 1 nM T99160 C71FQV 118598955 IC50 = 19 nM T99160 C48RSO 118598997 IC50 = 0.14 nM T99160 CCB0Q3 118599016 IC50 = 0.13 nM T99160 C4OZ3A 118599023 IC50 = 1.2 nM T99160 CJ4CB6 118599040 IC50 = 0.36 nM T99160 C6BEH9 118599128 IC50 = 2.6 nM T99160 CY7BI2 118706214 IC50 > 10000 nM T99160 CN0BQ3 118734651 Ki > 10000 nM T99160 C1U0RH 118734652 Ki > 10000 nM T99160 C1UTE7 118734653 Ki = 350 nM T99160 COK64U 118734654 Ki = 240 nM T99160 C6WQT5 118734655 Ki > 10000 nM T99160 C5ZD2P 118734656 Ki = 9050 nM T99160 C2LBN0 118734657 Ki = 5990 nM T99160 CIR0W7 118734658 Ki = 3170 nM T99160 CS6GO0 118734659 Ki = 2630 nM T99160 CJ5KP0 118734660 Ki = 340 nM T99160 C3CFZ7 118734661 Ki > 10000 nM T99160 CN0Z5J 118734662 Ki = 900 nM T99160 C7ZN0X 118734663 Ki = 1600 nM T99160 CC2T5L 121007996 IC50 = 1900 nM T99160 CC4P7E 122194697 Ki = 110 nM T99160 CH3BN2 122194698 Ki = 18 nM T99160 CGD5E3 122194699 Ki = 18 nM T99160 CYR1F2 122194700 Ki = 31 nM T99160 C7YMU6 122194701 Ki = 164 nM T99160 C8DW9G 122485490 IC50 = 1430 nM T99160 C4PFZ0 127046319 IC50 = 34 nM T99160 C0CX4P 127046320 IC50 = 2 nM T99160 CUD8G5 127046367 IC50 = 20 nM T99160 CA83YU 127047442 IC50 = 1 nM T99160 CNJQ71 127047443 IC50 = 0.7 nM T99160 CC1VO7 127047444 IC50 = 3 nM T99160 C3IRJ0 127048197 IC50 > 10000 nM T99160 CZ07TW 127048198 IC50 = 130 nM T99160 CS0H2C 127048199 IC50 > 10000 nM T99160 C1OE2F 127049532 IC50 = 8 nM T99160 C5P8TC 127049857 IC50 = 760 nM T99160 CPQ35R 127049870 IC50 = 10 nM T99160 CQO3X7 127049871 IC50 > 10000 nM T99160 C5H8LK 127051998 IC50 = 6860 nM T99160 CGT0B1 127052321 IC50 = 130 nM T99160 C7NH6A 127052914 IC50 = 1910 nM T99160 CKB1Y6 127052915 IC50 = 82 nM T99160 C3B8RF 129071308 IC50 = 45 nM T99160 CJ71ME 129071521 IC50 = 61 nM T99160 CZ5TU6 129071545 IC50 = 5.7 nM T99160 C1UWQ9 129956867 IC50 = 13000 nM T99160 C6OMB1 132204257 IC50 = 61 nM T99160 C0TA9U 134132267 IC50 < 1400 nM T99160 CJF28E 136273088 IC50 = 113 nM T99160 CXY09A 136621908 IC50 = 31 nM T99160 C4L5AY 136623815 IC50 = 140 nM T99160 C7SB9W 137652377 IC50 = 2700 nM T99160 C9ZO5R 137652825 IC50 = 7.8 nM T99160 C5G7EA 139307786 IC50 = 410 nM T99160 CXHK68 140999007 IC50 = 108000 nM T99160 CSG67A 141009064 IC50 = 171000 nM T99160 CL5F4T 141381328 IC50 = 415 nM T99160 CU65MQ 145915878 IC50 = 350 nM T99160 CNK29G 145949498 Ki = 110 nM T99160 C5JP4F 145949566 Ki = 2500 nM T99160 CGQ82M 145951244 Ki = 430 nM T99160 CW9U8I 145951798 Ki = 860 nM T99160 C0JB5Z 145951984 Ki = 560 nM T99160 CFV8U4 145952625 Ki = 120 nM T99160 CV8DJ4 145952962 Ki = 230 nM T99160 C0U5FM 145953025 Ki = 1570 nM T99160 CL6UR2 145953386 Ki = 1150 nM T99160 CU7I0F 145953845 Ki = 300 nM T99160 CM1XY4 145954013 Ki = 430 nM T99160 CESK62 145954175 Ki = 390 nM T99160 CMY39G 145956109 Ki = 610 nM T99160 CR8O6B 145956516 Ki = 200 nM T99160 C6D0NW 145956852 Ki = 220 nM T99160 CEM1D9 145957785 Ki = 1330 nM T99160 CE4VK8 145957843 Ki = 400 nM T99160 C95ORY 145958102 Ki = 1300 nM T99160 CH5SV6 145958167 Ki = 7700 nM T99160 CEK3W0 145958852 Ki = 180 nM T99160 C3N1XY 145959793 Ki = 110 nM T99160 C78BGW 145960126 Ki = 1700 nM T99160 CM8ZA1 145960224 Ki = 980 nM T99160 CXU0Z9 145964697 IC50 = 160 nM T99160 CR7HU3 145964902 IC50 = 515 nM T99160 C42FZC 145966011 IC50 = 193 nM T99160 C6O0GM 145972396 IC50 = 355 nM T99160 CGN0E7 145972578 IC50 = 742 nM T99160 C6NJ1Q 145976485 IC50 = 5170 nM T99160 CT4B8J 145977060 IC50 = 187 nM T99160 CE6R8H 145978647 IC50 = 1080 nM T99160 CWM5N2 145983960 IC50 = 1450 nM T99160 CN1A8H 145985334 IC50 = 273 nM T99160 CS4O6T 145985665 IC50 = 1160 nM T99160 CW4OT8 145985810 IC50 = 3550 nM T99160 C7U5OK 145986017 IC50 = 749 nM T99160 C9ME3Z 152452753 IC50 = 13000 nM T99160 C1SPV6 154726271 IC50 = 14 nM T99160 C2MD1Q 155513187 IC50 > 10000 nM T99160 CZUP45 155514353 IC50 = 120 nM T99160 C86ZGU 155515431 IC50 = 500 nM T99160 C3FH8B 155516612 IC50 = 44 nM T99160 CZB7S9 155520845 Ki = 82 nM T99160 CF19DM 155521087 IC50 = 340 nM T99160 C2P7HQ 155522861 IC50 = 410 nM T99160 CO5T8P 155523016 IC50 = 45000 nM T99160 CL9KF7 155523960 Ki = 1277 nM T99160 C9P5BJ 155525376 IC50 = 300 nM T99160 CT6PH0 155526131 IC50 = 160 nM T99160 C3EL4A 155526234 IC50 = 6900 nM T99160 C6DVW8 155528856 IC50 = 54 nM T99160 CBJ71H 155531160 IC50 = 390 nM T99160 CIO69B 155532028 Ki = 43 nM T99160 C8V7IT 155536337 IC50 = 730 nM T99160 CZOW93 155537061 IC50 = 5100 nM T99160 C52MTP 155537215 IC50 = 1400 nM T99160 C59FGZ 155541299 IC50 = 1200 nM T99160 CH7LV8 155545541 IC50 = 3000 nM T99160 CSY2X6 155545770 IC50 = 3300 nM T99160 C47TYE 155546525 IC50 = 7200 nM T99160 CKE71S 155548047 Ki = 438 nM T99160 C2OJ9K 155549245 IC50 = 460 nM T99160 CE4M8Y 155555762 IC50 = 6400 nM T99160 C94QIK 155557622 IC50 = 310 nM T99160 CB5NR2 155559630 IC50 = 1000 nM T99160 C1NVA6 155560651 IC50 = 16 nM T99160 CE6Y0J 155561742 IC50 = 1800 nM T99160 CGF1C5 155564109 IC50 = 970 nM T99160 CGH65C 155566572 IC50 = 80 nM T99160 CQ25XI 155566821 IC50 = 630 nM T99160 C37BGO 155567311 IC50 = 89 nM T99160 CYA3E9 155567459 IC50 = 42 nM T99160 C4AY9W 155568101 IC50 = 800 nM T99160 C8AOM4 11724428 IC50 = 450 nM T99160 D00ERW 44444843 Ki > 9350 nM T99160 D01KOI 346926 IC50 = 60000 nM T99160 D03DZO 11715767 IC50 = 171 nM T99160 D0A7FQ 11644425 Ki = 340 nM T99160 D0N7AJ 11409972 IC50 = 20 nM T99160 D0W6VA 82315 IC50 = 3700 nM T23172 D03ZBT 11626560 IC50 = 1360 nM T23172 D04LKS 25126798 Ki = 3.2 nM T23172 D04LVK 57379345 IC50 = 7920 nM T23172 D06XXH 11511120 IC50 = 3570000 nM T23172 D09KTS 24821094 IC50 = 22 nM T23172 D09XZB 123631 IC50 > 1000 nM T23172 D0EG1I 9926791 Ki = 0.24 nM T23172 D0Y7IC 44205240 IC50 = 25 nM T23172 D00RYA 16750271 IC50 = 4300 nM T23172 D00UZR 5330286 IC50 = 63.1 nM T23172 D02TUL 118115473 IC50 = 33 nM T23172 D03HUX 49792852 IC50 > 10000 nM T23172 D03LWG 53235510 IC50 > 10000 nM T23172 D04BFC 59174488 IC50 = 22.5 nM T23172 D04QWQ 59422203 Ki = 2.5 nM T23172 D05PCM 78323835 IC50 = 605 nM T23172 D05PZB 135398495 IC50 = 1 nM T23172 D06EIC 57928403 IC50 = 0.71 nM T23172 D06KTJ 53252276 IC50 = 114 nM T23172 D07EHV 44814409 IC50 > 10000 nM T23172 D07HPJ 11476171 IC50 > 10000 nM T23172 D07JAG 58557659 IC50 = 2300 nM T23172 D08HOM 46207586 IC50 > 10000 nM T23172 D0BI3N 44595079 IC50 = 8 nM T23172 D0D5ZJ 25062766 IC50 = 155 nM T23172 D0D8KQ 25127112 IC50 = 810 nM T23172 D0DK5X 135567296 IC50 = 59.9 nM T23172 D0DK8X 50922691 IC50 = 360 nM T23172 D0E3TC 44259 IC50 = 0.1 nM T23172 D0G5XV 135565884 IC50 = 580 nM T23172 D0G8BM 16722836 IC50 = 1000 nM T23172 D0H9FR 118295624 IC50 = 556 nM T23172 D0HS5V 11234052 IC50 > 50000 nM T23172 D0MP0X 16659841 IC50 = 1360 nM T23172 D0O0LS 25141092 IC50 = 349 nM T23172 D0PN8H 46216796 IC50 = 520 nM T23172 D0Q7RE 16007391 Ki > 10000 nM T23172 D0S1XX 134821691 IC50 > 10000 nM T23172 D0SG7B 49831257 IC50 = 810 nM T23172 D0VG0D 11977753 IC50 = 1000 nM T23172 D0YB3W 156414 IC50 = 2000 nM T23172 D0Y2PO 71770709 IC50 = 10500 nM T23172 D0T3ME 156422 IC50 > 30000 nM T23172 C8NW5J 3815 IC50 = 61 nM T23172 CRI78W 94391 IC50 > 100 nM T23172 C3F0GS 3120536 Ki > 5000 nM T23172 CGYE97 6419765 IC50 = 2000 nM T23172 C2OL7K 9796455 IC50 > 50000 nM T23172 CYA76E 9798589 IC50 > 100000 nM T23172 CRZ5T7 9815801 IC50 = 270 nM T23172 CYW49X 9927718 IC50 = 44 nM T23172 CQ89SE 9947841 IC50 = 27 nM T23172 C7YD1X 10048045 IC50 > 25000 nM T23172 CO70CQ 10107882 IC50 = 767 nM T23172 CP28QI 10154513 IC50 = 40 nM T23172 C35JMD 10269598 IC50 = 29 nM T23172 C7SFI1 10296883 IC50 = 1500 nM T23172 C2UWA0 10658651 IC50 = 710 nM T23172 CK2RY9 11164105 IC50 = 19 nM T23172 C2W5RC 11235063 IC50 > 50000 nM T23172 CBOP58 11293798 Ki > 10000 nM T23172 C26BZX 11362471 Ki > 10000 nM T23172 CWXB93 11397177 Ki > 10000 nM T23172 CT3VP7 11398307 IC50 = 25000000 nM T23172 CK83CN 11416425 IC50 = 7 nM T23172 CJC95A 11454205 IC50 > 10000 nM T23172 CU2OF8 11510392 IC50 = 557 nM T23172 C87ARG 11519208 IC50 = 37 nM T23172 CTG83F 11539329 Ki > 1700 nM T23172 C32PUD 11553058 IC50 = 140 nM T23172 CACS26 11561968 Ki = 1900 nM T23172 CI0X1C 11567474 IC50 = 1735 nM T23172 CMIL86 11590363 Ki > 1700 nM T23172 C45BMY 11603130 IC50 = 26 nM T23172 C69FYK 11604142 Ki = 280 nM T23172 CU6T2L 11613133 IC50 = 25 nM T23172 CG1JN5 11620467 IC50 = 110 nM T23172 C9ZD2E 11626406 IC50 = 1426 nM T23172 CK34LS 11632737 IC50 > 50000 nM T23172 C1TZY3 11635079 IC50 = 32 nM T23172 C9T6SC 11640926 Ki > 1700 nM T23172 CXG5W8 11646595 IC50 = 183 nM T23172 C3L2HT 11656560 IC50 = 1400 nM T23172 CX7C1T 11656606 IC50 = 71 nM T23172 C8RMT2 11663885 IC50 = 44 nM T23172 CP3U0W 11684933 IC50 = 960 nM T23172 CYO6X9 11684994 Ki = 6.5 nM T23172 CU0E8O 11690457 Ki = 280 nM T23172 CI3EO4 11692100 IC50 = 80 nM T23172 CB0AP2 11705863 Ki = 4800 nM T23172 CS36BH 11843159 IC50 = 1200 nM T23172 C61TIL 11844913 IC50 = 28 nM T23172 C9JT4S 11847343 IC50 = 3710 nM T23172 CHR92S 11858109 IC50 > 1000 nM T23172 CNYB84 11951225 IC50 = 28 nM T23172 C8E4TS 11992146 IC50 = 501.19 nM T23172 C58YUH 11993785 IC50 = 5.1 nM T23172 CW53JC 11998038 Ki = 3 nM T23172 C0Y7MG 12083227 IC50 = 160 nM T23172 CZI64D 12083230 IC50 = 390 nM T23172 C75SGK 12997800 IC50 = 77 nM T23172 CM9JA0 12997805 IC50 = 0.6 nM T23172 C47EVM 14487943 IC50 > 100 nM T23172 C9RQN8 15950748 IC50 > 25000 nM T23172 C0DUA7 15953425 IC50 = 3 nM T23172 C3JWA6 15953427 IC50 = 3 nM T23172 CWZM24 15953526 IC50 = 1.3 nM T23172 CSK90Y 15991573 IC50 = 20 nM T23172 CPNW35 15991575 IC50 > 8333 nM T23172 CFPW41 16007116 Ki > 1700 nM T23172 C12TIL 16058762 IC50 > 30000 nM T23172 C1WJ2D 16070041 IC50 > 10000 nM T23172 C3ZV2X 16086076 IC50 > 25000 nM T23172 C0SO7D 16086077 IC50 > 8333 nM T23172 C0WU9I 16086078 IC50 = 331 nM T23172 CVE6C8 16086088 IC50 = 16 nM T23172 CH1R8K 16086091 IC50 = 154 nM T23172 CT4RS8 16086092 IC50 = 1141 nM T23172 CZ2QU1 16086093 IC50 > 25000 nM T23172 C13OVU 16086099 IC50 = 133 nM T23172 C2YC0S 16086100 IC50 = 1339 nM T23172 C28UZX 16086101 IC50 > 8333 nM T23172 CKM8E4 16086102 IC50 = 16 nM T23172 CF0N4J 16086103 IC50 = 106 nM T23172 CKR57M 16086104 IC50 = 868 nM T23172 CI5HJ8 16086105 IC50 = 253 nM T23172 C68SBO 16086106 IC50 = 987 nM T23172 CAYV39 16086107 IC50 = 722 nM T23172 C06NOI 16086108 IC50 = 193 nM T23172 C16NRY 16086114 IC50 = 72 nM T23172 C87TPW 16086115 IC50 = 626 nM T23172 CW35LJ 16086116 IC50 = 2189 nM T23172 CA3BD7 16086117 IC50 > 25000 nM T23172 C3EKF4 16086118 IC50 > 8333 nM T23172 C0QCG4 16086142 IC50 = 46 nM T23172 CQG45C 16109001 IC50 = 25000 nM T23172 C1U8XW 16109036 IC50 = 1700 nM T23172 CZ5Y3V 16116847 IC50 > 25000 nM T23172 CLO43V 16116849 IC50 > 25000 nM T23172 C0HO6T 16118191 IC50 > 25000 nM T23172 CT92BZ 16118192 IC50 > 25000 nM T23172 CIZ6B4 16118193 IC50 > 25000 nM T23172 C2CN5O 16118323 IC50 > 25000 nM T23172 C4GTU3 16118324 IC50 > 25000 nM T23172 CXC78K 16118603 IC50 > 25000 nM T23172 CI4E6Y 16118605 IC50 > 25000 nM T23172 C8LIW4 16118609 IC50 > 25000 nM T23172 CGC34R 16118737 IC50 > 25000 nM T23172 CAN2K6 16118739 IC50 > 25000 nM T23172 CT8WS0 16126645 IC50 = 45 nM T23172 C5VPH9 16129448 IC50 = 496 nM T23172 CI83KB 16216717 IC50 = 3 nM T23172 CM32VW 16659676 IC50 = 2960 nM T23172 CO3L1Q 16659677 IC50 = 200 nM T23172 CL38VY 16659680 IC50 = 8350 nM T23172 C0ECA7 16659682 IC50 > 30000 nM T23172 CXYV28 16659836 IC50 = 5250 nM T23172 C91SVD 16659838 IC50 = 30 nM T23172 CC10IO 16662069 IC50 = 30500 nM T23172 CD1NT2 16662070 IC50 > 30000 nM T23172 C19KHB 16664854 IC50 = 142 nM T23172 CO7E8C 16678106 IC50 > 5000 nM T23172 CY1E2N 16723801 IC50 = 52000 nM T23172 C0H8UN 16730109 IC50 > 50000 nM T23172 CSE35D 16739464 IC50 > 10000 nM T23172 C20OFQ 16739508 IC50 > 10000 nM T23172 CCP56J 16739905 IC50 > 10000 nM T23172 CQ64XI 16739921 IC50 > 10000 nM T23172 CM3UF8 16739935 IC50 > 10000 nM T23172 CFEP56 16739948 IC50 > 10000 nM T23172 C23KZR 16739951 IC50 > 10000 nM T23172 C9OQ1G 16750272 IC50 > 10000 nM T23172 CW2SY5 16750291 IC50 = 650 nM T23172 CIX7U2 16750304 IC50 = 8800 nM T23172 C6A3XS 16750306 IC50 = 680 nM T23172 CB2TK1 16750327 IC50 = 9200 nM T23172 CH4O1C 16750328 IC50 = 1000 nM T23172 C90MJD 16750331 IC50 > 10000 nM T23172 C7JW2E 18008439 IC50 = 210 nM T23172 C24XMR 19917815 IC50 = 142 nM T23172 CG31WF 20111936 IC50 = 43 nM T23172 C6UAZ0 20820292 IC50 = 3250 nM T23172 C87BYV 22282847 IC50 = 143 nM T23172 CJ5GR1 22282945 IC50 = 117 nM T23172 C50FBN 22282953 IC50 = 147 nM T23172 CO5WJ8 22484447 IC50 = 65 nM T23172 C16TAZ 22484511 IC50 = 370 nM T23172 COW73Q 22484526 IC50 = 138 nM T23172 CE7K3W 23532567 IC50 > 10000 nM T23172 CD7M2U 23582566 IC50 = 6800 nM T23172 CUY98W 23585560 IC50 = 18 nM T23172 C5Y1QX 23644715 IC50 = 213 nM T23172 C7YG1N 24759534 IC50 = 280 nM T23172 CAJ4T2 24762205 IC50 > 10000 nM T23172 CQNP54 24764449 IC50 = 1000 nM T23172 C4Z9CN 24769780 IC50 > 25000 nM T23172 CLBP72 24798571 IC50 = 528 nM T23172 CX1U4S 24800423 IC50 > 10000 nM T23172 C4T0DG 24800602 IC50 > 10000 nM T23172 CH3ZG7 24800604 IC50 > 10000 nM T23172 CBA02Y 24800776 IC50 = 670 nM T23172 C3UFG1 24801129 IC50 = 130 nM T23172 CVR8S1 24801650 IC50 = 450 nM T23172 CYBI02 24823426 IC50 > 25000 nM T23172 C45UGH 24823586 IC50 = 438 nM T23172 CFA3T8 24823588 IC50 > 25000 nM T23172 C51ZTV 24823589 IC50 > 25000 nM T23172 CX0QC1 24823590 IC50 > 25000 nM T23172 CR7CH6 24823736 IC50 > 25000 nM T23172 C26KXV 24823738 IC50 > 25000 nM T23172 CO3K7R 24823740 IC50 > 5000 nM T23172 CBLJ48 24823898 IC50 > 25000 nM T23172 CG0K1Z 24824046 IC50 > 25000 nM T23172 C59FKG 24860777 IC50 > 10000 nM T23172 CL0O9E 24877325 IC50 > 980 nM T23172 CY0P4X 24877326 IC50 > 980 nM T23172 C7R4YV 24877438 IC50 > 980 nM T23172 C5G4BY 24877439 IC50 > 980 nM T23172 C5NXH3 24877440 IC50 > 980 nM T23172 CJ4Z0K 24877791 IC50 = 104.5 nM T23172 CQUH61 24877795 IC50 > 980 nM T23172 CO5RV2 24878018 IC50 > 980 nM T23172 CH3Q1D 24878130 IC50 > 980 nM T23172 C4MG3B 24882476 IC50 = 334 nM T23172 CY8L7E 24896769 IC50 > 10000 nM T23172 CWV98O 24899557 IC50 > 10000 nM T23172 C5S7XA 24958852 IC50 = 5.2 nM T23172 CJ68PR 24958855 IC50 = 9.2 nM T23172 CZ18IU 24963047 IC50 = 2930 nM T23172 CBK82P 25011729 IC50 = 20500 nM T23172 CT07ZW 25030805 IC50 = 229 nM T23172 CHLC27 25052652 IC50 > 30000 nM T23172 C7W6FX 25059112 IC50 = 85 nM T23172 CD0T4Z 25059626 IC50 = 274 nM T23172 CD4TJ7 25059891 IC50 = 2020 nM T23172 CE9N8F 25060146 IC50 = 66 nM T23172 C3Y7SB 25060677 IC50 = 2310 nM T23172 CWZH04 25060922 IC50 = 192 nM T23172 C7VPB2 25060927 IC50 = 9 nM T23172 C25NMK 25061435 IC50 = 1450 nM T23172 CF3Z0Q 25061949 IC50 = 1876 nM T23172 CF3QE4 25061950 IC50 = 3910 nM T23172 C2BEQ3 25062226 IC50 > 1000 nM T23172 CSVH95 25062228 IC50 = 1760 nM T23172 C9KY0J 25062498 IC50 > 1000 nM T23172 CG4U2Y 25062765 IC50 > 5000 nM T23172 CVI87D 25063021 IC50 = 364 nM T23172 C4JO2C 25063023 IC50 = 1418 nM T23172 C3VIR1 25063025 IC50 = 362 nM T23172 CF9X4L 25069658 IC50 = 39 nM T23172 C5Q4KO 25069976 IC50 = 5 nM T23172 C0H4SC 25070616 IC50 = 72 nM T23172 CP1W7D 25070617 IC50 = 17.5 nM T23172 C0X4NG 25070618 IC50 = 36 nM T23172 CJDZ19 25070619 IC50 = 27 nM T23172 CNQ07G 25103042 IC50 = 262 nM T23172 C09PMH 25103279 IC50 = 20 nM T23172 C1V7QM 25103281 IC50 = 30 nM T23172 COP15B 25103284 IC50 = 15 nM T23172 CP8GU7 25104502 IC50 = 95 nM T23172 C7EK6V 25104503 IC50 = 262 nM T23172 C63ADF 25104611 IC50 = 11230 nM T23172 CON1U6 25110598 IC50 = 763 nM T23172 C0JYA9 25123154 IC50 = 2500 nM T23172 C56JVD 25123155 IC50 = 1300 nM T23172 CZM6Q2 25123472 IC50 = 280 nM T23172 C3IA7V 25123474 IC50 > 10000 nM T23172 C6V4NB 25123475 IC50 = 1500 nM T23172 CFK89A 25123806 IC50 = 360 nM T23172 C3RMN9 25123807 IC50 = 4900 nM T23172 C5GO3T 25123808 IC50 = 8300 nM T23172 C0W8IC 25124143 IC50 = 1350 nM T23172 C61WOA 25127137 IC50 = 5200 nM T23172 C4WFL0 25128110 IC50 = 1300 nM T23172 CFK46X 25138051 IC50 = 98 nM T23172 C4M2XQ 25138052 IC50 = 2640 nM T23172 CQMU82 25138148 IC50 = 156 nM T23172 CD9O6K 25138149 IC50 = 3040 nM T23172 COV8Z0 25143021 IC50 > 10000 nM T23172 CI0E2L 25154395 IC50 = 1400 nM T23172 CL1W5D 25154436 IC50 = 1000 nM T23172 CSO82D 25154877 Ki = 170 nM T23172 C8GL6I 25169133 IC50 = 12730 nM T23172 C1G5JU 25169403 IC50 > 30000 nM T23172 CZ28ES 25171661 IC50 = 13730 nM T23172 C6ZTG4 25171663 IC50 = 11710 nM T23172 CQ04LW 25171665 IC50 = 5030 nM T23172 CU9KV5 25171666 IC50 = 5170 nM T23172 C0SE7H 25171874 IC50 = 25050 nM T23172 C1YH8L 25171876 IC50 = 26880 nM T23172 CC60NT 25171877 IC50 = 15220 nM T23172 C8O1ZJ 25172085 IC50 = 12770 nM T23172 CG6J5X 25172086 IC50 = 3660 nM T23172 CRO8T9 25263033 Ki > 12500 nM T23172 CC71QJ 27666048 IC50 > 100000 nM T23172 CY4LG8 42622934 IC50 = 300 nM T23172 C57VJY 42635854 IC50 = 230 nM T23172 CP8RA7 42635855 IC50 = 220 nM T23172 C05BWT 42635901 IC50 = 220 nM T23172 CO9Y8F 42635906 IC50 = 740 nM T23172 CN1TI5 42635944 IC50 = 140 nM T23172 C5I9XW 42635949 IC50 = 170 nM T23172 CT63QC 42635982 IC50 = 210 nM T23172 CY5E4B 42635983 IC50 = 280 nM T23172 C8V6IK 42635984 IC50 = 220 nM T23172 C63HQD 42636016 IC50 = 270 nM T23172 C34DCR 42636018 IC50 = 370 nM T23172 CTOQ08 42636019 IC50 = 160 nM T23172 CU8MO6 42641406 IC50 = 54 nM T23172 CCB1E9 44124695 IC50 > 100000 nM T23172 CQI60M 44158549 IC50 = 11000 nM T23172 CBAN65 44158553 IC50 = 240 nM T23172 CH6OL2 44158658 IC50 = 86 nM T23172 CHD5N8 44158660 IC50 = 180 nM T23172 CU07NR 44158886 IC50 = 200 nM T23172 CLK7R8 44159000 IC50 = 10 nM T23172 CD0YP3 44159001 IC50 = 12 nM T23172 CQ8FJ4 44159590 IC50 = 39 nM T23172 CY67LR 44159594 IC50 = 17 nM T23172 CZF1B5 44159711 IC50 = 25 nM T23172 CQW4F1 44159839 IC50 = 230 nM T23172 CBK83A 44159959 IC50 = 160 nM T23172 CEF0X4 44159962 IC50 = 49 nM T23172 CBZ09W 44160079 IC50 = 4400 nM T23172 C1ZY4N 44160207 IC50 = 7 nM T23172 CIT2A7 44192904 IC50 = 17 nM T23172 C8KNA3 44219632 Ki > 4000 nM T23172 C0VIX4 44219633 Ki = 2300 nM T23172 C9WO8E 44335773 IC50 = 26 nM T23172 C1GZO3 44335832 IC50 = 260 nM T23172 CM9EG2 44335843 IC50 = 200 nM T23172 C75JOK 44335848 IC50 = 350 nM T23172 C7EVL3 44335849 IC50 = 235 nM T23172 C5AIE1 44335857 IC50 = 30 nM T23172 C1QSC2 44335927 IC50 = 7100 nM T23172 CT39UY 44335938 IC50 = 190 nM T23172 C7HLB8 44335946 IC50 = 4900 nM T23172 CP04EM 44335947 IC50 = 2300 nM T23172 CV0JK5 44335968 IC50 = 168 nM T23172 CUA46C 44335985 IC50 = 210 nM T23172 C8U9PJ 44335986 IC50 = 870 nM T23172 C4R0CG 44336174 IC50 = 700 nM T23172 CZB49P 44419474 IC50 = 61 nM T23172 CI9GX4 44419475 IC50 = 27 nM T23172 CAT2U0 44419478 IC50 = 120 nM T23172 CC36WM 44419481 IC50 = 131 nM T23172 C6BWA2 44419485 IC50 = 180 nM T23172 CXW0D5 44419491 IC50 = 21 nM T23172 CZY28V 44419492 IC50 = 92 nM T23172 CCM3W5 44419493 IC50 = 60 nM T23172 CG2R1T 44419498 IC50 = 1928 nM T23172 C40WFE 44419499 IC50 = 860 nM T23172 CNZJ15 44419502 IC50 = 62 nM T23172 C5DL8E 44419515 IC50 > 10000 nM T23172 CMVY72 44419516 IC50 = 470 nM T23172 CNT03L 44419522 IC50 = 9097 nM T23172 CH46CM 44419523 IC50 = 700 nM T23172 CO20LA 44419524 IC50 = 49 nM T23172 C3CBQ4 44419526 IC50 = 145 nM T23172 C4XIY6 44419527 IC50 > 10000 nM T23172 CGH30Q 44419528 IC50 = 245 nM T23172 C42FJP 44419532 IC50 > 10000 nM T23172 C0FKV6 44419533 IC50 = 42 nM T23172 CXG7H4 44419544 IC50 = 167 nM T23172 CI2BL7 44419547 IC50 = 51 nM T23172 C2T5AQ 44419548 IC50 = 31 nM T23172 CT19AN 44419556 IC50 = 83 nM T23172 CE6T5F 44419559 IC50 = 19 nM T23172 CBH85Y 44430889 IC50 = 13.5 nM T23172 CQ46MX 44430894 IC50 = 3 nM T23172 C6EXR2 44430895 IC50 = 80 nM T23172 CW5AF1 44430896 IC50 = 250 nM T23172 C0KQN7 44430897 IC50 = 23.5 nM T23172 CVY2R6 44430898 IC50 = 15 nM T23172 CDYE48 44430900 IC50 = 70 nM T23172 CJ8EH7 44430901 IC50 = 3130 nM T23172 C2D1TN 44430902 IC50 = 14 nM T23172 CFIE13 44430903 IC50 = 1050 nM T23172 CSA7N0 44430904 IC50 > 5000 nM T23172 C9OT6G 44430905 IC50 = 354 nM T23172 C07EGM 44430907 IC50 = 592 nM T23172 CARH16 44430909 IC50 = 109 nM T23172 CWY7Z5 44430910 IC50 = 11 nM T23172 C3B1ME 44430911 IC50 = 31 nM T23172 C70KJQ 44430914 IC50 = 686 nM T23172 CF90PO 44430915 IC50 = 237 nM T23172 CQ0Y6P 44432177 IC50 = 22 nM T23172 CSRD60 44432179 IC50 = 18 nM T23172 C1DZ5C 44432180 IC50 = 34 nM T23172 CWBI39 44432182 IC50 = 42 nM T23172 C73SGA 44432183 IC50 = 46 nM T23172 CA92GM 44432184 IC50 = 49 nM T23172 CTDI23 44432185 IC50 = 67 nM T23172 CI9NY3 44432187 IC50 = 77 nM T23172 CGFT15 44432188 IC50 = 126 nM T23172 CT0D6O 44432189 IC50 = 142 nM T23172 CFK94T 44432190 IC50 = 143 nM T23172 C3TG1J 44432191 IC50 = 200 nM T23172 CBO5P0 44432192 IC50 = 430 nM T23172 C2S8ZC 44432193 IC50 = 3050 nM T23172 CUB12D 44449577 IC50 > 50000 nM T23172 CDV6X9 44454507 IC50 > 25000 nM T23172 C6SMY7 44454538 IC50 > 25000 nM T23172 CZI92T 44454651 IC50 > 25000 nM T23172 CIA39D 44454676 IC50 > 25000 nM T23172 C7DGA2 44454678 IC50 > 25000 nM T23172 C1F3LT 44454702 IC50 > 25000 nM T23172 CCW57R 44454703 IC50 > 25000 nM T23172 CFS7W2 44454728 IC50 > 25000 nM T23172 CTL43P 44454729 IC50 > 25000 nM T23172 CZC95J 44454731 IC50 > 25000 nM T23172 CYH6P3 44520205 IC50 = 8140 nM T23172 C3XTA7 44562721 Ki = 74 nM T23172 C5YL2S 44570390 IC50 = 370 nM T23172 C63WNF 44610370 IC50 > 30000 nM T23172 CT7V9E 44610371 IC50 = 28500 nM T23172 CL40ZN 44610523 IC50 > 30000 nM T23172 C6QT0J 44622837 IC50 > 1000 nM T23172 CU3RF1 45139989 IC50 > 10000 nM T23172 CQGZ06 45139991 IC50 > 10000 nM T23172 CY83PR 45267327 IC50 = 1 nM T23172 CRXU30 45269072 IC50 > 200 nM T23172 C84QFJ 45269074 IC50 = 6 nM T23172 C1S0PJ 45269930 IC50 = 9 nM T23172 CDJZ52 45271570 IC50 = 8 nM T23172 C7PNR2 45272482 IC50 = 9 nM T23172 CB1C9W 45272486 IC50 = 12 nM T23172 CIE14V 45273357 IC50 = 3 nM T23172 C3DH8I 45273358 IC50 = 7 nM T23172 CHK79Y 45273361 IC50 = 15 nM T23172 CO5QA1 45273364 IC50 = 39 nM T23172 C4J5XF 45275254 IC50 = 3930 nM T23172 CZ7T8F 45275363 IC50 = 1440 nM T23172 CB58EO 45275368 IC50 = 7560 nM T23172 CU3AD0 45275473 IC50 = 1820 nM T23172 C7KMO9 45275580 IC50 = 14830 nM T23172 C96HCQ 45375954 IC50 = 15 nM T23172 CQ3KO2 45375955 IC50 = 1.7 nM T23172 C5G2MN 45375956 IC50 = 1 nM T23172 C6OX0V 45375974 IC50 = 26480 nM T23172 CXF92W 45486106 IC50 = 2100 nM T23172 CZXL23 45486109 IC50 = 460 nM T23172 CF8JM7 45486113 IC50 = 190 nM T23172 CIE6V0 45486118 IC50 = 500 nM T23172 CV59GT 45486119 IC50 = 2100 nM T23172 C9E0MS 45486120 IC50 = 220 nM T23172 C07DPA 45486121 IC50 = 170 nM T23172 CR7T9D 45486124 IC50 = 1600 nM T23172 C7QK0X 45486129 IC50 = 4000 nM T23172 CY36ZX 45486130 IC50 = 420 nM T23172 C04ZHY 45486136 IC50 > 30000 nM T23172 C5SA2N 45486137 IC50 = 1800 nM T23172 C91VMT 45486138 IC50 = 210 nM T23172 CLN7F0 45486139 IC50 = 67 nM T23172 C8RNJ5 45486142 IC50 = 12 nM T23172 C9FQJ4 45486147 IC50 = 600 nM T23172 CPM6O9 45486148 IC50 = 570 nM T23172 CX0HO6 45486156 IC50 = 15670 nM T23172 CYZ13M 45486157 IC50 > 30000 nM T23172 CZMD28 45486158 IC50 = 2800 nM T23172 CMXY69 45486159 IC50 = 200 nM T23172 CA0O3Q 45486163 IC50 = 210 nM T23172 C5U1LS 45486164 Ki = 400 nM T23172 CN6G7A 45486168 IC50 > 30000 nM T23172 CT9OP5 45486169 IC50 > 30000 nM T23172 C7D4GB 45486170 IC50 = 290 nM T23172 CE45XW 46208354 IC50 = 0.46 nM T23172 CUHB49 46208355 IC50 = 0.72 nM T23172 CW38GO 46208357 IC50 = 0.61 nM T23172 C43COY 46208358 IC50 = 0.36 nM T23172 CE4Q7D 46208596 IC50 = 1.1 nM T23172 CM9UN7 46208601 IC50 = 0.39 nM T23172 CH7JB4 46209051 IC50 = 0.8 nM T23172 CZ58FY 46215814 IC50 = 990 nM T23172 CY3HW5 46224684 IC50 = 5300 nM T23172 C7ON5A 46233287 IC50 > 10000 nM T23172 CG6Y3N 46234403 IC50 = 1083 nM T23172 C3JW8A 46234405 IC50 > 1000 nM T23172 CWN3M0 46234565 IC50 = 22 nM T23172 CLTU68 46234566 IC50 = 10 nM T23172 C5YH1F 46235625 IC50 = 268 nM T23172 CWLU63 46235938 IC50 = 695 nM T23172 CC25DT 46235942 IC50 = 29 nM T23172 CZ7J6K 46236109 IC50 = 20 nM T23172 C26NQY 46236112 IC50 = 82 nM T23172 C1S4LH 46398810 IC50 = 610 nM T23172 C35AIH 46865430 IC50 = 190 nM T23172 C2EK4B 46865431 IC50 = 160 nM T23172 CMZ0R3 46865529 IC50 = 166 nM T23172 C3B2NL 46865530 IC50 = 230 nM T23172 CC2O9R 46865656 IC50 = 1995.26 nM T23172 CLS29B 46872626 IC50 > 10000 nM T23172 C0AU7R 46879420 IC50 = 6 nM T23172 CUVG95 46879421 IC50 = 220 nM T23172 CRZM17 46879422 IC50 = 95 nM T23172 CER6X5 46879423 IC50 = 48 nM T23172 C7O1AZ 46879483 IC50 = 365 nM T23172 C2DU1O 46879484 IC50 = 260 nM T23172 CB31AL 46879485 IC50 = 30 nM T23172 C5URZ1 46879545 IC50 = 170 nM T23172 C3LEW4 46879546 IC50 = 540 nM T23172 CKI4M6 46880119 IC50 = 115 nM T23172 CU8KB7 46880120 IC50 = 245 nM T23172 C47OXF 46880121 IC50 = 68 nM T23172 CK87XC 46880122 IC50 = 38 nM T23172 CC3Y7B 46880193 IC50 = 14 nM T23172 C0GS1C 46880194 IC50 = 7 nM T23172 CV9IL3 46880195 IC50 = 108 nM T23172 C0M5ND 46880196 IC50 = 17 nM T23172 C60UAN 46880197 IC50 = 70 nM T23172 C5NZ8R 46880686 IC50 = 2000 nM T23172 CZ79VE 46880687 IC50 = 400 nM T23172 CGO7C5 46880738 IC50 = 300 nM T23172 C75ZTG 46880739 IC50 = 620 nM T23172 C9T7WL 46880784 IC50 = 170 nM T23172 CSV4G2 46880785 IC50 = 220 nM T23172 C6Z4KW 46882470 IC50 = 110 nM T23172 CH0Y5K 46882471 IC50 = 538 nM T23172 C70LVA 46882472 IC50 = 930 nM T23172 CP1BH3 46882539 IC50 = 636 nM T23172 CQR25C 46882540 IC50 > 1000 nM T23172 CVTO81 46882541 IC50 = 1619 nM T23172 CQ6T0Y 46882542 IC50 = 960 nM T23172 COV4E6 46882589 IC50 > 1000 nM T23172 CDG2N8 46882590 IC50 = 587 nM T23172 C0UX2M 46882591 IC50 = 351 nM T23172 CN0I6Z 46882592 IC50 = 149 nM T23172 CZ7A9N 46882802 IC50 = 364 nM T23172 CCK7H2 46882803 IC50 = 152 nM T23172 C9MW2L 46885052 IC50 > 10000 nM T23172 C69HUW 46885053 IC50 > 10000 nM T23172 CASL67 46885231 IC50 = 2700 nM T23172 CEU6O4 46885232 IC50 = 9900 nM T23172 CE27LI 46885233 IC50 = 232 nM T23172 CB8LN4 46885234 IC50 = 408 nM T23172 CMX7U6 46885289 IC50 = 630 nM T23172 CB1ZN5 46885290 IC50 = 130 nM T23172 C2O8RZ 46886323 IC50 > 1000 nM T23172 C60GAV 46929544 IC50 > 8000 nM T23172 CP34VL 46929748 IC50 > 1000 nM T23172 CJ2E9Q 46929857 IC50 > 25000 nM T23172 CCN08S 46934144 IC50 = 34200 nM T23172 CT7EY8 49817363 IC50 = 27 nM T23172 CBP75U 49838138 IC50 = 17 nM T23172 CMKB24 49838268 IC50 = 31 nM T23172 CF0UM2 49838516 IC50 = 39 nM T23172 CTJX98 49838518 IC50 = 89 nM T23172 CSE4K3 49838775 IC50 = 38 nM T23172 C9L3XR 49838879 IC50 > 10000 nM T23172 C06MKW 49839561 Ki = 253 nM T23172 CT3SH4 49839838 IC50 = 286 nM T23172 CF91RS 49843531 IC50 > 10000 nM T23172 C4LM3X 49855554 IC50 = 2 nM T23172 C9UZ6E 49855558 IC50 = 210 nM T23172 CR6Q5Y 49855559 IC50 = 350 nM T23172 CTM0I6 49855750 IC50 = 110 nM T23172 CJXR91 49855751 IC50 = 58 nM T23172 CXH97G 49855752 IC50 = 20 nM T23172 CXN17D 49855753 IC50 = 61 nM T23172 CC5LP1 49855941 IC50 = 230 nM T23172 C8V3HY 49855942 IC50 = 540 nM T23172 C4V8AF 49856128 IC50 = 20 nM T23172 CS3Q7G 49856129 IC50 = 32 nM T23172 CM2V5K 49856130 IC50 = 38 nM T23172 CHZ58U 49856131 IC50 = 13 nM T23172 C8NI4M 49856317 IC50 = 150 nM T23172 C57FQH 49856318 IC50 = 14 nM T23172 C70QSD 49856319 IC50 = 26 nM T23172 C24SMN 49856320 IC50 = 42 nM T23172 CHK7D3 49856321 IC50 = 32 nM T23172 C2XIV5 49856322 IC50 = 480 nM T23172 CY6JH3 49856512 IC50 = 230 nM T23172 CQ6OG4 49856516 IC50 = 39 nM T23172 C90VXM 49856700 IC50 = 20 nM T23172 CK4LJ5 49856703 Ki = 120 nM T23172 CA0WR3 50914031 IC50 = 57 nM T23172 CQE9D1 50925411 IC50 = 1 nM T23172 C2Y6QS 50938552 IC50 > 10000 nM T23172 CF26MU 50991562 IC50 = 3800 nM T23172 CHS63D 50993724 IC50 = 4590 nM T23172 C2SKV4 50993725 IC50 > 30000 nM T23172 CKN2H7 50993726 IC50 > 30000 nM T23172 CMH3A2 50993881 IC50 = 11800 nM T23172 C20VEP 50994284 IC50 > 10000 nM T23172 CI1L0M 50994285 IC50 = 133 nM T23172 C7ZWT8 50994286 IC50 = 423 nM T23172 C6VNE1 50994366 IC50 = 36 nM T23172 CSEZ73 50994367 IC50 = 460 nM T23172 C1R8ZI 50995341 IC50 = 17 nM T23172 C53NRD 50995522 IC50 = 15 nM T23172 C9NYP4 51036677 IC50 > 10000 nM T23172 C4WRY3 51037112 IC50 > 10000 nM T23172 CRI28Z 51037948 IC50 > 10000 nM T23172 CEQN27 52936621 Ki = 350 nM T23172 CM24LF 52938983 IC50 < 1 nM T23172 CA9DE6 52941228 IC50 > 10000 nM T23172 C1T5EH 52942437 IC50 > 10000 nM T23172 CEPS91 52943663 IC50 = 2000 nM T23172 C2IQ5B 52943672 IC50 > 10000 nM T23172 CTN0C3 52944839 IC50 > 10000 nM T23172 CAB1Y3 52946772 IC50 > 100 nM T23172 CT2U3E 52947304 IC50 = 1250 nM T23172 CQY9D0 52948526 IC50 = 1470 nM T23172 C8TC3P 52948550 IC50 = 850 nM T23172 CIM43G 52948562 IC50 = 5000 nM T23172 CR36JQ 53232414 IC50 = 349.1 nM T23172 C93WOC 53232452 IC50 = 21 nM T23172 CH3Y2L 53317729 IC50 = 18000 nM T23172 CL14DA 53317826 IC50 = 13 nM T23172 C72DMQ 53320251 IC50 = 113 nM T23172 CZM72A 53320461 IC50 = 4 nM T23172 C82DGQ 53321752 IC50 = 2000 nM T23172 CHFX17 53321753 IC50 = 1200 nM T23172 CTBJ21 53322914 IC50 = 800 nM T23172 C2W9OA 53324451 IC50 > 10000 nM T23172 CZKQ72 53341161 Ki = 369 nM T23172 CB83XH 53341368 Ki = 130 nM T23172 CGP23R 53341457 Ki = 3.8 nM T23172 C8ZRE3 53356518 IC50 = 33740 nM T23172 C8NA4L 53384644 IC50 > 30000 nM T23172 C56TYK 53385837 IC50 = 48.5 nM T23172 CNLM53 53385838 IC50 = 68.9 nM T23172 C1XE2K 53385938 IC50 = 148 nM T23172 C37JTE 53385939 IC50 = 8.2 nM T23172 CV92IB 53386254 IC50 = 5.2 nM T23172 CU6QF7 53386309 IC50 < 0.4 nM T23172 CYU0R4 53386418 IC50 = 0.44 nM T23172 C7RM6Q 53386421 IC50 < 0.3 nM T23172 CEN91X 53389820 IC50 = 104.4 nM T23172 C37PHN 53497571 IC50 = 1340 nM T23172 CCF1B3 53497572 IC50 = 307 nM T23172 COG24D 53820179 IC50 > 100 nM T23172 CY5C8A 54589404 IC50 = 0.26 nM T23172 CS7E0A 54672927 IC50 = 44.5 nM T23172 CHZ27O 54673255 IC50 = 8.6 nM T23172 C7X5ZM 54673258 IC50 = 9.6 nM T23172 CZ84NW 54673259 IC50 = 1.4 nM T23172 CX0U2A 54673422 IC50 = 7.8 nM T23172 C19FZK 54673425 IC50 = 43.6 nM T23172 CBPT15 54673763 IC50 = 140 nM T23172 C36BAI 54673911 IC50 = 1.8 nM T23172 CD8ZK6 54674056 IC50 = 30 nM T23172 CFTE97 54674369 IC50 = 210 nM T23172 CUCI05 54674990 IC50 = 19 nM T23172 CH0IM9 54754557 IC50 = 2.7 nM T23172 C1XS2J 54760383 IC50 = 2600 nM T23172 CXH2P4 54766274 IC50 = 34 nM T23172 CD28VZ 54766423 IC50 = 53 nM T23172 CAP1J7 54766425 IC50 = 260 nM T23172 C75JFM 54766426 IC50 = 490 nM T23172 CDIC43 54766427 IC50 = 59 nM T23172 C2XDG1 54766428 IC50 = 80 nM T23172 C0XCY1 54766576 IC50 = 96 nM T23172 CPH3Y7 54766578 IC50 = 47 nM T23172 C0T4SL 54766726 IC50 = 39 nM T23172 CZD70Q 54767039 IC50 = 4.9 nM T23172 CN1DZ6 54767189 IC50 = 8.4 nM T23172 C1W3EZ 56591424 IC50 = 3.9 nM T23172 CTB63S 56591428 IC50 = 64 nM T23172 CWR1P6 56591446 IC50 = 1 nM T23172 C6ZL7H 56592816 IC50 = 80 nM T23172 C6Z1QA 56592817 IC50 = 2.6 nM T23172 CKZ27O 56594916 IC50 = 1900 nM T23172 CR70XD 56595052 IC50 = 560 nM T23172 C3DJO1 56595053 IC50 = 1700 nM T23172 C8KO5T 56595054 IC50 = 640 nM T23172 CW4QC9 56595056 IC50 = 430 nM T23172 CM8JX1 56604907 IC50 = 10000 nM T23172 C1FA3D 56659205 IC50 = 720 nM T23172 CY1QA2 56683053 IC50 = 350 nM T23172 CR9A5O 56834874 IC50 = 3330 nM T23172 C58MSV 56834889 IC50 = 963 nM T23172 CUT2G8 56835062 IC50 = 2.9 nM T23172 CBFR12 56925356 IC50 = 967 nM T23172 C80DRA 56925357 IC50 = 2870 nM T23172 C0HUN8 56925358 IC50 > 125000 nM T23172 C6Z2EA 56925359 IC50 = 10300 nM T23172 CC1MN2 56925454 IC50 = 1660 nM T23172 C3XC0T 56925455 IC50 = 545 nM T23172 CBW6T3 56925456 IC50 = 188 nM T23172 C8G3NO 56925457 IC50 = 365 nM T23172 CHS19C 56925458 IC50 = 118 nM T23172 CBMO42 56925459 IC50 = 434 nM T23172 CQTD41 56925550 IC50 = 1280 nM T23172 CI9T3S 56925551 IC50 = 2380 nM T23172 CS84ZU 56925552 IC50 = 645 nM T23172 C9IVD0 56929216 Ki = 22 nM T23172 CSO40C 56973425 Ki = 33 nM T23172 CU5BD9 57336812 IC50 = 150 nM T23172 CPO2J4 57342178 IC50 > 10000 nM T23172 C72PED 57342179 IC50 = 1140 nM T23172 CA93PN 57342180 IC50 > 10000 nM T23172 CZSM95 57412684 IC50 > 10000 nM T23172 C6A8WC 57502370 IC50 > 3000 nM T23172 CIO15D 57502371 IC50 > 10000 nM T23172 C6YOU9 57502372 IC50 > 10000 nM T23172 C8DN1A 57502373 IC50 > 10000 nM T23172 C15XOS 57502374 IC50 > 10000 nM T23172 CEF53Z 57502376 IC50 > 2000 nM T23172 CTY54N 57502377 IC50 = 834 nM T23172 CBLN61 57502378 IC50 = 475 nM T23172 CDV4R1 57502379 IC50 = 95 nM T23172 CILJ54 57502380 IC50 > 10000 nM T23172 CS90RX 57502381 IC50 = 63 nM T23172 CE6B7C 57502382 IC50 = 31 nM T23172 CC82QJ 57502383 IC50 = 146 nM T23172 C72OWZ 57502386 IC50 = 60 nM T23172 CHC90Q 57502387 IC50 = 122 nM T23172 C9Z6QJ 57502388 IC50 = 72 nM T23172 CMF31G 57502390 IC50 = 547 nM T23172 C4QXU9 57514090 IC50 > 3000 nM T23172 C0YW2D 57514091 IC50 = 598 nM T23172 CU8Y3P 57514092 IC50 = 105 nM T23172 C5K3VZ 57514093 IC50 = 218 nM T23172 COU4M1 57915982 IC50 = 28 nM T23172 C1G5SK 57916044 IC50 = 22 nM T23172 C3C0PQ 57916049 IC50 = 54 nM T23172 CH6RB0 57916164 IC50 = 42 nM T23172 C9MF8U 57928260 IC50 = 2.1 nM T23172 C3KQJ8 57928435 IC50 = 0.43 nM T23172 C5H8VE 57928583 IC50 = 2.1 nM T23172 C13VIO 57928632 IC50 = 10 nM T23172 C8BTO7 57928826 IC50 = 0.63 nM T23172 C18MVX 57990771 IC50 = 5000 nM T23172 C4TQ9L 57990797 IC50 = 368.1 nM T23172 C4XC3V 57990957 IC50 > 980 nM T23172 CB6F5S 57990969 IC50 = 61.7 nM T23172 CDRB84 57991074 IC50 > 980 nM T23172 CJ4B2L 57991089 IC50 = 159.8 nM T23172 C9EA1S 57991186 IC50 = 557.3 nM T23172 C48LZT 57991260 IC50 > 980 nM T23172 C8R4FE 57991377 IC50 = 214.2 nM T23172 C19UKS 57991389 IC50 = 483.8 nM T23172 C1KH5D 57991398 IC50 = 306.8 nM T23172 CSN47V 57991473 IC50 = 298.3 nM T23172 CQND09 58177229 IC50 = 18 nM T23172 CU4I8X 58177247 IC50 = 18 nM T23172 CLEH36 58177279 IC50 = 8 nM T23172 CIK3U8 58177332 IC50 = 27 nM T23172 C8D2TA 58177362 IC50 = 37 nM T23172 CYC85B 58177456 IC50 = 1 nM T23172 C7BU0H 58180518 IC50 = 49 nM T23172 CKA28H 58180521 IC50 = 87 nM T23172 C2I5LO 58180525 IC50 = 77 nM T23172 CN4OZ8 58180573 IC50 = 460 nM T23172 C92FOB 58180591 IC50 = 19 nM T23172 CWXC70 58180596 IC50 = 160 nM T23172 C9N1QB 58180623 IC50 = 210 nM T23172 CSK1U8 58180628 IC50 = 62 nM T23172 C6LT9S 58180630 IC50 = 23 nM T23172 CCBT87 58180639 IC50 = 52 nM T23172 CP81TW 58394456 Ki = 200 nM T23172 C0F3BO 58394783 Ki = 110 nM T23172 CO5TH6 58394820 Ki = 220 nM T23172 C0X7IK 58394837 Ki = 280 nM T23172 C9Q4WD 58394916 Ki = 130 nM T23172 CASI81 58395078 Ki = 5.9 nM T23172 CDK5L1 58395223 Ki = 24 nM T23172 CWBM72 58395283 Ki = 7.8 nM T23172 C9TV2G 58398904 IC50 = 30000 nM T23172 CR9T7W 58438557 IC50 = 8.7 nM T23172 CY3W6B 58438580 IC50 = 80.6 nM T23172 CR7C4V 58438607 IC50 = 0.4 nM T23172 C9MIL7 58450666 IC50 = 4.5 nM T23172 CWX4G9 58522116 IC50 = 1380 nM T23172 C4A6LT 58522124 IC50 = 340 nM T23172 CI9VB0 58522237 IC50 = 370 nM T23172 C1LE9A 58522238 IC50 = 420 nM T23172 C74ACR 58522276 IC50 = 400 nM T23172 CI0L1J 58522322 IC50 = 470 nM T23172 CVMO97 58522377 IC50 = 970 nM T23172 C7S1PR 58522381 IC50 = 280 nM T23172 C1SI3L 59174579 IC50 = 1533 nM T23172 CPWM60 59291925 IC50 = 1.2 nM T23172 C3CV0R 59291929 IC50 = 25 nM T23172 COXI75 59291940 IC50 = 25 nM T23172 CE6KO4 59291951 IC50 = 1.7 nM T23172 CT3EW2 59292007 IC50 = 0.3 nM T23172 C2PE0T 59292008 IC50 = 3.6 nM T23172 CU3W2S 59292043 IC50 = 3.4 nM T23172 CC6J4I 59363349 IC50 = 7 nM T23172 CQ93TM 59363383 IC50 = 2 nM T23172 CKQ31B 59363409 IC50 = 5 nM T23172 CXJ63M 59603829 IC50 = 430 nM T23172 CQEU96 59603842 IC50 = 33 nM T23172 COH62U 60097413 IC50 > 5000 nM T23172 C1MR8Q 60097495 IC50 > 5000 nM T23172 CNY59P 60165955 Ki = 0.9 nM T23172 CY3QT8 60165956 Ki = 22 nM T23172 CJ08ZL 66604045 IC50 = 193 nM T23172 CY0I2V 66604274 IC50 = 264 nM T23172 CD0LJ6 66604359 IC50 = 139 nM T23172 CS8HK2 66604394 IC50 = 48 nM T23172 C7U8GC 66604464 IC50 = 311 nM T23172 CXU94O 66604576 IC50 = 123 nM T23172 CE9T0V 66604664 IC50 = 2021 nM T23172 C7WO4A 66604791 IC50 = 59 nM T23172 CW53KR 66604810 IC50 = 324 nM T23172 CNW05G 66604855 IC50 = 119 nM T23172 C0JS8O 66604914 IC50 = 35 nM T23172 CW9LD1 66604921 IC50 = 130 nM T23172 CTMX20 66605009 IC50 = 246 nM T23172 CP0DB1 66605115 IC50 = 59 nM T23172 CB1WC9 66605298 IC50 = 225 nM T23172 CCWU74 66605322 IC50 = 66 nM T23172 C7Q8ZG 66605359 IC50 = 990 nM T23172 C16TEK 66605475 IC50 = 442 nM T23172 C7MOJ6 66605487 IC50 = 197 nM T23172 CDZA70 66605639 IC50 = 242 nM T23172 C53NBQ 66605756 IC50 = 66 nM T23172 C5PVB2 67008690 IC50 = 14 nM T23172 C8OZ6W 67008828 IC50 = 22 nM T23172 C1HSE0 67035086 IC50 = 7200 nM T23172 CWI6K5 67035106 IC50 > 10000 nM T23172 C38RGB 67035556 IC50 > 10000 nM T23172 CZX1E0 67123420 IC50 = 420 nM T23172 C0RCI2 67123577 IC50 = 3 nM T23172 C37NKO 67129970 IC50 > 10000 nM T23172 CK80LJ 67130050 IC50 > 10000 nM T23172 CV63UL 67240318 IC50 > 10000 nM T23172 C6YHJ5 67277266 IC50 = 240 nM T23172 C78TXA 67277273 IC50 = 46 nM T23172 C0O7TC 67277276 IC50 = 1.1 nM T23172 C3YK7Q 67277763 IC50 = 90 nM T23172 CQXW93 67277840 IC50 = 460 nM T23172 CF4AB0 67277979 IC50 = 1100 nM T23172 CFM39N 67278030 IC50 = 340 nM T23172 C5U2IW 67278045 IC50 = 21 nM T23172 CS9K0L 67278047 IC50 = 710 nM T23172 C2FW8H 67278142 IC50 = 69 nM T23172 CQRS42 67278151 IC50 = 63 nM T23172 C5V9DZ 67278165 IC50 = 270 nM T23172 CMJ29W 67278195 IC50 = 60 nM T23172 C2C7BD 67278380 IC50 = 150 nM T23172 CVL35U 67278385 IC50 = 180 nM T23172 CKVB79 67278425 IC50 = 27 nM T23172 CV80IQ 67330694 IC50 = 2460 nM T23172 CKMV48 67345882 Ki = 76 nM T23172 CFX84K 67352945 Ki = 122 nM T23172 C9WY2P 67383875 Ki = 58 nM T23172 C5WQC2 67502257 IC50 = 1 nM T23172 CYR38C 68241014 IC50 = 22 nM T23172 CW23JE 68241353 IC50 = 7 nM T23172 C0MY1I 68241371 IC50 = 25 nM T23172 CCBA10 68241463 IC50 = 37 nM T23172 CX6S4E 68254533 IC50 > 30000 nM T23172 C4U1IR 68291322 IC50 = 6 nM T23172 C2P7DB 68291391 IC50 = 32 nM T23172 CRM3S0 68291627 IC50 = 43 nM T23172 C4LKB3 68291752 IC50 = 1 nM T23172 CQ49HB 68291755 IC50 = 3 nM T23172 CXI4L1 68291797 IC50 = 24 nM T23172 C8T5VB 68291830 IC50 = 5 nM T23172 CPRW18 68291866 IC50 = 14 nM T23172 C6UWI3 68291981 IC50 = 12 nM T23172 CYN89R 68292156 IC50 = 67 nM T23172 C76EZC 68292170 IC50 = 16 nM T23172 CGA0W6 68292183 IC50 = 10 nM T23172 C93LZT 68292196 IC50 = 47 nM T23172 C8I7GC 68293638 IC50 > 10000 nM T23172 CD56XK 68293660 IC50 > 10000 nM T23172 CYI75G 68678653 IC50 > 30000 nM T23172 C7GRV2 68755406 IC50 > 10000 nM T23172 CIL58T 69023801 IC50 = 1149.3 nM T23172 C5DGR9 69036886 IC50 = 3162 nM T23172 CK8DC3 69046862 IC50 = 3.2 nM T23172 CV0K3P 69267827 IC50 = 87 nM T23172 COX56A 69809432 IC50 = 10 nM T23172 CECG39 69809726 IC50 = 20 nM T23172 C7FA5L 69811602 IC50 = 2 nM T23172 C92EAC 69811936 IC50 = 5 nM T23172 C0XO1M 69812740 IC50 = 31 nM T23172 CASQ98 70650259 IC50 = 49 nM T23172 CNR2Y9 71061323 IC50 = 1.1 nM T23172 C51JTW 71061588 IC50 = 3.6 nM T23172 CF69WT 71061828 IC50 = 0.7 nM T23172 COU2C5 71061858 IC50 = 18 nM T23172 CW9OE6 71061878 IC50 = 1.4 nM T23172 CK9LZ3 71061981 IC50 = 2.4 nM T23172 CU1T4P 71061987 IC50 = 40 nM T23172 CJH94D 71062030 IC50 = 3.5 nM T23172 CUW46K 71062043 IC50 = 3.4 nM T23172 C05VNE 71062076 IC50 = 6 nM T23172 C4AC9U 71212257 IC50 = 12 nM T23172 C7Y2LB 71230234 Ki = 53 nM T23172 COR71Z 71285696 IC50 = 0.6 nM T23172 C3ZL5S 71285760 IC50 = 1.8 nM T23172 CME92O 71285933 IC50 = 3.1 nM T23172 C2FL6H 71286084 IC50 = 0.8 nM T23172 C14YOJ 71286184 IC50 = 10 nM T23172 CX23BP 71288497 IC50 = 2.9 nM T23172 CH1AJ3 71288512 IC50 = 0.3 nM T23172 CA1T5H 71288539 IC50 = 1.8 nM T23172 CYU2Z4 71288594 IC50 = 3 nM T23172 CBY4K0 71288602 IC50 = 1.1 nM T23172 CWLC45 71288607 IC50 = 2.3 nM T23172 CDST08 71288618 IC50 = 1 nM T23172 C45HTF 71288693 IC50 = 0.8 nM T23172 COC20B 71288707 IC50 = 10.5 nM T23172 C6JD3S 71288724 IC50 < 0.4 nM T23172 COV78A 71288729 IC50 = 0.3 nM T23172 C8DY1N 71288732 IC50 = 3.4 nM T23172 CNV7B6 71300296 IC50 = 20 nM T23172 CKT60L 71455860 Ki > 1700 nM T23172 C4D1TQ 71456076 IC50 > 980 nM T23172 CCN01X 71547862 IC50 > 10000 nM T23172 CVIA91 71553085 IC50 = 30000 nM T23172 C1TR3O 71553152 IC50 = 30000 nM T23172 CVEO06 71558636 IC50 = 5 nM T23172 C1SR5V 71576693 IC50 = 175 nM T23172 C07SFW 71600166 IC50 = 112 nM T23172 CWJ1G4 71600167 IC50 = 57 nM T23172 CKY79O 71615499 IC50 = 8 nM T23172 C8GLY0 71615500 IC50 = 45 nM T23172 CA7Q3S 71615501 IC50 = 4 nM T23172 CVYS15 71617859 IC50 = 2.8 nM T23172 CS62NH 71698376 IC50 = 78.12 nM T23172 CI8X1R 71698379 IC50 = 418.2 nM T23172 C5QK6S 71727668 IC50 = 41 nM T23172 C4X1CP 71748056 IC50 = 3336 nM T23172 CKO8S6 71815907 IC50 = 343 nM T23172 C54XWG 72190869 IC50 > 10000 nM T23172 CLD12K 72201823 IC50 = 153.1 nM T23172 CYQN46 72201826 IC50 = 56.7 nM T23172 CP9CJ3 72201957 IC50 = 500.5 nM T23172 CMVI93 72201958 IC50 = 204.2 nM T23172 CD9Z4H 72202092 IC50 = 195.1 nM T23172 CLIS85 72202093 IC50 = 178.1 nM T23172 C5Q7YT 72202095 IC50 = 5083 nM T23172 C8NGE4 72202097 IC50 = 226.1 nM T23172 C1W6LK 72202246 IC50 = 175.8 nM T23172 C6W4ZS 72202247 IC50 = 88.1 nM T23172 C1N7LQ 72202249 IC50 = 7.6 nM T23172 C2W6TI 72202397 IC50 = 33.7 nM T23172 CIKL36 72202398 IC50 = 52 nM T23172 C1I4LX 72202399 IC50 = 140.5 nM T23172 C4CB2S 72202400 IC50 = 136.1 nM T23172 CVI63X 72202547 IC50 = 12 nM T23172 C0EZ3I 72202548 IC50 = 94.7 nM T23172 C7OY3V 72202549 IC50 = 274.9 nM T23172 CH40KC 72202550 IC50 = 95.7 nM T23172 CIU90H 72202607 IC50 = 7100 nM T23172 CA5CI3 72202825 IC50 = 32.4 nM T23172 CK7F6U 72700776 Ki = 37 nM T23172 CLOE10 72706962 IC50 = 54 nM T23172 C9OQ2I 72710839 IC50 > 10000 nM T23172 C4BUW7 73353407 IC50 = 16400 nM T23172 CF6QG1 73602845 IC50 = 983 nM T23172 CDN83F 73707530 IC50 = 38.1 nM T23172 CCQN01 73775788 IC50 = 25.3 nM T23172 CHF08G 73775789 IC50 = 218 nM T23172 COL37D 73775921 IC50 > 10000 nM T23172 CVQW20 73775923 IC50 = 650 nM T23172 C5U4AF 73776059 IC50 = 192 nM T23172 CXW54V 73776061 IC50 = 177 nM T23172 CD83FL 73776204 IC50 = 38.6 nM T23172 CG84BR 73776205 IC50 = 17.4 nM T23172 C1P3DO 73776206 IC50 = 1520 nM T23172 CN5D1R 73776207 IC50 = 5640 nM T23172 CO1C8Y 73776208 IC50 = 2150 nM T23172 CGC46K 73776360 IC50 = 983 nM T23172 C8DSE2 75108379 IC50 = 5880 nM T23172 CS41CX 75108409 IC50 = 3780 nM T23172 CH20VA 75108447 IC50 = 13150 nM T23172 CP90QE 75108517 IC50 > 30000 nM T23172 CG6T5S 76072368 IC50 = 23.2 nM T23172 COMF95 76072369 IC50 = 91.3 nM T23172 CO0BQ5 76310565 IC50 = 13 nM T23172 C6ZAB2 76310566 IC50 > 10000 nM T23172 C0F6VU 76310567 IC50 = 128 nM T23172 CDO38G 76310568 IC50 > 10000 nM T23172 CL42BQ 76310569 IC50 = 163 nM T23172 CWI1Q4 76310570 IC50 = 12 nM T23172 C8OY6Q 76310785 IC50 > 100000 nM T23172 CAL3U7 76310788 IC50 > 100000 nM T23172 C7SXJ1 76314208 IC50 = 135 nM T23172 CSDI71 76314209 IC50 = 46 nM T23172 CY61RI 76314210 IC50 = 408 nM T23172 CO2M7V 76314211 IC50 = 1387 nM T23172 C12YAE 76314414 IC50 > 100000 nM T23172 CXF1I3 76317774 IC50 = 497 nM T23172 CY79VS 76317775 IC50 > 10000 nM T23172 CNK2I1 76317776 IC50 = 278 nM T23172 CS02NA 76317777 IC50 = 179 nM T23172 CAHW32 76317778 IC50 = 625 nM T23172 CT9JM4 76317888 IC50 > 30000 nM T23172 C97RBS 76317979 IC50 > 100000 nM T23172 C2SMK1 76321491 IC50 > 10000 nM T23172 C2DSX7 76321492 IC50 = 200 nM T23172 CXA4O1 76325093 IC50 = 9367 nM T23172 CEZ64F 76325209 IC50 = 4620 nM T23172 C1AI0J 76325315 IC50 > 100000 nM T23172 CPQA45 76325323 IC50 > 100000 nM T23172 C8GK0H 76328659 IC50 = 576 nM T23172 C0WK6O 76328660 IC50 = 1499 nM T23172 CJN89E 76332335 IC50 = 1790 nM T23172 CW1QK4 76332336 IC50 = 29 nM T23172 CFX05K 76332337 IC50 = 1380 nM T23172 C2P1MX 76332338 IC50 = 576 nM T23172 CB5Y0Z 76332540 IC50 > 100000 nM T23172 CJ2T9E 76332983 IC50 > 10000 nM T23172 CB4KQ7 76335967 IC50 = 1148 nM T23172 C84PFQ 76335968 IC50 = 201 nM T23172 CW1HQ9 76370451 IC50 = 0.71 nM T23172 CD6Y1F 78320046 IC50 >= 8000 nM T23172 CW08SU 78320048 IC50 >= 8000 nM T23172 CWI93D 78323836 IC50 >= 8000 nM T23172 C5UK9L 78323837 IC50 >= 8000 nM T23172 CQ3EJ1 78324132 IC50 >= 8000 nM T23172 C7VOX0 78324136 IC50 >= 8000 nM T23172 CA2Y8L 78324435 IC50 >= 8000 nM T23172 C4I7WD 78324744 IC50 >= 8000 nM T23172 CN39OQ 78341183 IC50 = 49 nM T23172 CQ2SU8 78673832 IC50 > 30000 nM T23172 CE0W9R 78673833 IC50 > 30000 nM T23172 CPG3A5 86302574 IC50 > 30000 nM T23172 C96EDF 86660048 IC50 = 3400 nM T23172 CC8I0M 86707711 IC50 = 0.9 nM T23172 CW4Z2F 89470642 IC50 = 230 nM T23172 CBRF87 89470690 IC50 = 511 nM T23172 C7B8OH 89470730 IC50 = 100 nM T23172 CDQ8C6 89471114 IC50 = 256 nM T23172 C4G5LP 89471136 IC50 = 361 nM T23172 CW2RX5 89629876 IC50 = 0.15 nM T23172 CS7GX8 89708625 IC50 = 478.1 nM T23172 C1HW4B 89735655 IC50 = 1300 nM T23172 CG9C6J 89765129 IC50 = 31 nM T23172 C13GOX 89775209 IC50 = 52 nM T23172 C3N6RU 89775221 IC50 = 6.4 nM T23172 CI5WT1 90001694 IC50 > 5000 nM T23172 CTV52A 90367281 IC50 = 1226 nM T23172 CY0UC4 90645194 IC50 > 10000 nM T23172 C7EXH8 91755097 IC50 = 0.6 nM T23172 C37IZB 91755098 IC50 = 6.1 nM T23172 C7UAK5 91809175 IC50 > 2000 nM T23172 C8RG6H 91827514 IC50 = 1400 nM T23172 CVR1I7 91827515 IC50 = 230 nM T23172 C64SIO 92042864 IC50 = 4.8 nM T23172 C9BL4M 92045136 IC50 = 8300 nM T23172 CAKD54 102594000 IC50 > 10000 nM T23172 CM2C3W 105539869 IC50 = 82 nM T23172 CU4O5Z 112901888 IC50 = 2100 nM T23172 C3ECY5 117625437 IC50 = 2.8 nM T23172 CZC84D 117769161 IC50 = 2.1 nM T23172 CE7BZ8 117769174 IC50 = 11 nM T23172 CBJ07Q 117769217 IC50 = 4.6 nM T23172 CXHQ08 117769229 IC50 = 0.4 nM T23172 CS9WO4 117769234 IC50 = 0.9 nM T23172 C61VXQ 117769241 IC50 = 0.8 nM T23172 C1SA9I 117769244 IC50 = 0.4 nM T23172 C0VY7C 117769271 IC50 = 1.3 nM T23172 C6O9BT 117769272 IC50 = 3.8 nM T23172 CSR9B0 117769289 IC50 = 0.5 nM T23172 C2M9CR 117769307 IC50 = 1.6 nM T23172 C7FWS3 117769309 IC50 = 1 nM T23172 CYWV32 117769339 IC50 = 1 nM T23172 CZV35K 117769346 IC50 = 1.6 nM T23172 C5V6RG 117769349 IC50 = 6.7 nM T23172 C4O1PX 117769362 IC50 = 1.6 nM T23172 CPV4C8 117769365 IC50 = 1.5 nM T23172 CP3MC5 117769379 IC50 = 1.5 nM T23172 C8V6LG 117769392 IC50 = 0.9 nM T23172 C2NBZ8 117769396 IC50 = 1 nM T23172 COV59Y 117769408 IC50 = 1.8 nM T23172 CXJ3I6 117769409 IC50 = 1.1 nM T23172 C8LTZ6 117769464 IC50 = 4 nM T23172 C4KL1Y 117769470 IC50 = 0.7 nM T23172 CQ46WT 117769476 IC50 = 2.8 nM T23172 CSKO30 117769533 IC50 = 1.9 nM T23172 C6XC3W 117769575 IC50 = 0.9 nM T23172 CS95HO 117769592 IC50 = 1.3 nM T23172 C0PIL5 117769623 IC50 = 1.9 nM T23172 CO3DA2 117769866 IC50 = 23 nM T23172 CI46CP 117770056 IC50 = 100 nM T23172 C7NI8L 117770083 IC50 = 85 nM T23172 CJ3QC8 117770200 IC50 = 2200 nM T23172 CSD47C 117770482 IC50 = 5.3 nM T23172 C8SNB9 117770595 IC50 = 39 nM T23172 CJ1V9A 117770654 IC50 = 27 nM T23172 CS8E6M 117770678 IC50 = 1900 nM T23172 CM7X9N 117770754 IC50 = 32 nM T23172 C4CFG6 117770831 IC50 = 92 nM T23172 C0X1EQ 117809257 IC50 = 3 nM T23172 CDUH09 117809287 IC50 = 0.6 nM T23172 C8HYU9 117926195 IC50 > 10000 nM T23172 CRU03Y 118115411 IC50 > 10000 nM T23172 CGQK96 118115537 IC50 = 0.4 nM T23172 CI1V2B 118115600 IC50 = 56 nM T23172 CRS83F 118115605 IC50 > 10000 nM T23172 CO8I5F 118115659 IC50 > 10000 nM T23172 C2OX1Q 118115706 IC50 = 75 nM T23172 C2ZM7V 118115718 IC50 = 60 nM T23172 CKB13H 118115831 IC50 > 10000 nM T23172 CWCO47 118115913 IC50 = 1610 nM T23172 C20WGT 118115950 IC50 = 2021 nM T23172 C72LYV 118116131 IC50 = 0.7 nM T23172 CB3LR2 118116220 IC50 > 2478 nM T23172 CN5QT8 118116221 IC50 = 7570 nM T23172 C4JW5D 118116385 IC50 = 3840 nM T23172 CJGT03 118346182 IC50 = 5580 nM T23172 C02DGP 118346184 IC50 = 1560 nM T23172 CU6NE2 118346192 IC50 = 654 nM T23172 CW25VP 118346194 IC50 = 224 nM T23172 C4D2ZP 118475611 IC50 = 0.87 nM T23172 C1MV6H 118475615 IC50 = 83 nM T23172 C3PL4C 118475617 IC50 = 0.7 nM T23172 CQEL95 118475618 IC50 = 0.7 nM T23172 CF6I1Z 118475620 IC50 = 2.9 nM T23172 CK6Z8O 118475621 IC50 = 0.6 nM T23172 C7U4BT 118475622 IC50 = 1.2 nM T23172 C1PT9V 118475623 IC50 < 0.5 nM T23172 C4SR5G 118475624 IC50 = 4.4 nM T23172 CC79KI 118475625 IC50 < 0.5 nM T23172 C96ONC 118475626 IC50 = 0.58 nM T23172 C0AYV7 118475628 IC50 = 31 nM T23172 CJI4D6 118475629 IC50 = 245 nM T23172 CH8T1S 118475632 IC50 = 3.6 nM T23172 C89VQM 118475634 IC50 = 1.1 nM T23172 CEW97C 118475635 IC50 < 0.5 nM T23172 C9Z4QV 118475637 IC50 < 0.5 nM T23172 C4L6YH 118475642 IC50 = 1.7 nM T23172 CYE0M8 118475643 IC50 = 1.4 nM T23172 CIVS69 118475644 IC50 < 0.5 nM T23172 CLGD78 118475645 IC50 = 2720 nM T23172 CK9OX1 118475646 IC50 = 1.4 nM T23172 CW3N7P 118475647 IC50 < 0.5 nM T23172 CU1LX2 118475648 IC50 = 1.2 nM T23172 C17FYA 118475649 IC50 = 20 nM T23172 CG95ZB 118475650 IC50 = 7.4 nM T23172 C0VYQ4 118475651 IC50 = 6.2 nM T23172 CE49ZI 118475652 IC50 < 0.5 nM T23172 CB93OQ 118475653 IC50 = 0.6 nM T23172 C2V3ZW 118475655 IC50 = 0.6 nM T23172 CXQ7E5 118475656 IC50 < 0.5 nM T23172 C5JL0G 118475657 IC50 = 0.7 nM T23172 C65NIK 118475658 IC50 = 12.3 nM T23172 CO90AT 118475660 IC50 = 30 nM T23172 C75WLA 118475662 IC50 = 390 nM T23172 CEWP08 118475663 IC50 = 7 nM T23172 C5MOB2 118475664 IC50 = 222 nM T23172 CWJI73 118475666 IC50 = 31 nM T23172 CC3F6J 118475667 IC50 = 0.9 nM T23172 CI8D3B 118475668 IC50 = 0.9 nM T23172 CWH8V2 118475670 IC50 = 499 nM T23172 CFOX06 118475671 IC50 = 99 nM T23172 C5J9KB 118475672 IC50 = 46 nM T23172 CH3BE2 118475673 IC50 = 20 nM T23172 COQ1E3 118475674 IC50 = 0.5 nM T23172 CRQ5W2 118475675 IC50 = 4.6 nM T23172 CX60YK 118475676 IC50 = 1.6 nM T23172 C2D1IJ 118475677 IC50 < 0.5 nM T23172 CO25DM 118475692 IC50 = 2570 nM T23172 C71FOS 118475704 IC50 = 18 nM T23172 C0A9RJ 118475705 IC50 = 1.3 nM T23172 C4G7DS 118475713 IC50 = 170 nM T23172 C3W2LG 118475714 IC50 = 2.3 nM T23172 C0E6FR 118475715 IC50 = 12 nM T23172 CK3S8I 118475721 IC50 = 1600 nM T23172 C0M1NY 118475723 IC50 = 0.7 nM T23172 C31DBL 118475724 IC50 = 6.6 nM T23172 CX3N2U 118475727 IC50 = 64 nM T23172 CWQ38Z 118475750 IC50 = 258 nM T23172 CG3Q9J 118475753 IC50 = 24 nM T23172 CC13YD 118475754 IC50 = 0.9 nM T23172 CE3X0Q 118475759 IC50 = 2 nM T23172 CWQ36P 118475893 IC50 = 7.9 nM T23172 CN04RH 118475894 IC50 = 2.1 nM T23172 CGM29Q 118475901 IC50 = 101 nM T23172 C2P0CG 118475938 IC50 = 2.3 nM T23172 CEA5U1 118475940 IC50 = 17 nM T23172 CJYV54 118494221 IC50 = 21.8 nM T23172 CLTV08 118690376 IC50 = 3.3 nM T23172 CRK6J2 118690573 IC50 = 4 nM T23172 CTR74C 118690690 IC50 = 4.6 nM T23172 C3Z6GN 118705186 IC50 = 0.43 nM T23172 CY7BI2 118706214 IC50 > 10000 nM T23172 C2C0AG 118707521 IC50 > 100000 nM T23172 C2DJA0 118707522 IC50 > 100000 nM T23172 CBF28W 118707523 IC50 > 100000 nM T23172 CQ6ON4 118707525 IC50 > 100000 nM T23172 C38UWP 118707526 IC50 > 100000 nM T23172 C64ZQX 118707543 IC50 > 100000 nM T23172 CX58DI 118716791 IC50 > 30000 nM T23172 CD9X2B 118716796 IC50 > 30000 nM T23172 C2YJ0O 118716797 IC50 > 30000 nM T23172 CL3UO9 118716798 IC50 > 30000 nM T23172 C71BAM 118716799 IC50 > 30000 nM T23172 CU4EL6 118716806 IC50 > 30000 nM T23172 CP0IO9 118722564 IC50 = 334 nM T23172 C5K2QD 118723914 IC50 = 8 nM T23172 C59YJC 118723915 IC50 = 5 nM T23172 C2ON7Y 118723916 IC50 = 110 nM T23172 C5U8WG 118723917 IC50 = 66 nM T23172 C0ZMR8 118723918 IC50 = 28 nM T23172 C4Z5LJ 118723919 IC50 = 30 nM T23172 C85ELI 118723920 IC50 = 15 nM T23172 CGW49X 118723921 IC50 = 69 nM T23172 CXC8K9 118723922 IC50 = 42 nM T23172 CR5JD8 118723923 IC50 = 24 nM T23172 C9W1BU 118723924 IC50 = 140 nM T23172 C8JGN7 118868847 IC50 >= 8000 nM T23172 C3DK1Q 118868914 IC50 >= 8000 nM T23172 CQ1TL7 118879520 IC50 = 219 nM T23172 C5Z0XH 118911481 IC50 = 1100 nM T23172 CT4MJ8 118911570 IC50 = 110 nM T23172 C37DUM 121293882 IC50 = 28 nM T23172 CXQR89 121294143 IC50 = 11 nM T23172 CO7D4I 122182021 IC50 = 1200 nM T23172 CY9M5S 122182022 IC50 = 5 nM T23172 C2MCH6 122182157 IC50 = 23 nM T23172 CD92SA 122182158 IC50 = 130 nM T23172 CK4A6L 122182159 IC50 = 0.78 nM T23172 C1DUI6 122184730 IC50 = 0.6 nM T23172 CW4OC3 122184731 IC50 = 7.8 nM T23172 C1KWA0 122184792 IC50 = 5.2 nM T23172 CA17NI 122185109 IC50 = 2 nM T23172 CW3UH0 122185110 IC50 = 1.3 nM T23172 CC7GN4 122185111 IC50 = 220 nM T23172 C9OWX5 122186256 IC50 > 10000 nM T23172 C3J6BA 122186261 IC50 > 10000 nM T23172 CZN2V0 122188510 IC50 = 3068 nM T23172 CD62MC 122191616 IC50 = 130 nM T23172 CJI3E4 122191617 IC50 = 510 nM T23172 CFU15S 122191618 IC50 = 190 nM T23172 CE4F3A 122191619 IC50 > 2000 nM T23172 CAC5U1 122191620 IC50 = 500 nM T23172 C8C1PI 122191621 IC50 = 200 nM T23172 CA0D5W 122191622 IC50 = 2900 nM T23172 CZ9K5C 122191623 IC50 = 670 nM T23172 C3NYR0 122191624 IC50 = 5800 nM T23172 CRF2K0 122191625 IC50 = 5000 nM T23172 CPY1K9 122191778 IC50 = 35 nM T23172 C1H4IX 122192065 IC50 = 1500 nM T23172 C98EJO 122192066 IC50 = 1800 nM T23172 CM1XD7 122192067 IC50 = 1500 nM T23172 C0MLH5 122192068 IC50 = 1100 nM T23172 CC4T6A 122192069 IC50 = 1260 nM T23172 CGO6M7 122192070 IC50 = 2500 nM T23172 CBP34K 122192071 IC50 = 14100 nM T23172 CA2TF6 122192072 IC50 = 2100 nM T23172 CFY30Z 122192073 IC50 = 1900 nM T23172 CJ09XF 122192074 IC50 = 2300 nM T23172 C6LS8X 122192075 IC50 = 1900 nM T23172 C7DJA5 122192076 IC50 = 2100 nM T23172 CAS86F 122192079 IC50 = 10500 nM T23172 CG7TP0 122192080 IC50 = 1900 nM T23172 C5K8UM 122192081 IC50 = 2500 nM T23172 C4X7SD 122192466 IC50 > 10000 nM T23172 CS4XB9 122199230 IC50 >= 8000 nM T23172 CNA45R 122362931 IC50 = 22 nM T23172 C98UIX 122362933 IC50 = 470 nM T23172 CW5VJ4 122362934 IC50 = 548 nM T23172 C4AXS0 122362935 IC50 = 226 nM T23172 C6JO4C 122474157 IC50 = 67.1 nM T23172 C0XB2E 122475292 IC50 > 100 nM T23172 CLM7K3 122604539 IC50 > 10000 nM T23172 C01JHI 122604566 IC50 > 10000 nM T23172 C9QCD3 126715362 IC50 > 30000 nM T23172 CNPB25 126715363 IC50 > 30000 nM T23172 CJS53A 126715367 IC50 > 30000 nM T23172 CX37RN 126715380 IC50 > 30000 nM T23172 C2DQU9 126715387 IC50 > 30000 nM T23172 C1QB5R 126715400 IC50 = 19100 nM T23172 CG7YQ2 126715454 IC50 > 30000 nM T23172 CR9C1G 127030133 IC50 > 1400 nM T23172 CU4AJ8 127037981 IC50 > 30000 nM T23172 CA0O1B 127037982 IC50 > 30000 nM T23172 C50NKB 127037983 IC50 > 30000 nM T23172 CF8KQ6 127038326 IC50 > 30000 nM T23172 C5WV8P 127038327 IC50 = 27600 nM T23172 CI8ZB6 127038328 IC50 > 30000 nM T23172 C98DQZ 127038947 IC50 = 7470 nM T23172 CQ4OE5 127039917 IC50 > 30000 nM T23172 CC1XP0 127040339 IC50 > 22000 nM T23172 C8H7JN 127040340 IC50 = 19200 nM T23172 CRQS46 127040341 IC50 > 30000 nM T23172 C3B0AP 127040342 IC50 > 30000 nM T23172 C7KLD9 127040660 IC50 = 4500 nM T23172 C4JF8H 127040661 IC50 = 1200 nM T23172 CC9J7R 127040662 IC50 = 6900 nM T23172 CP1RY4 127040993 IC50 = 1540 nM T23172 C7P5MY 127040994 IC50 = 6140 nM T23172 CB23SC 127041238 IC50 = 16900 nM T23172 CJ7QW5 127041248 IC50 > 30000 nM T23172 C1N6BC 127041249 IC50 = 6600 nM T23172 C5SLH0 127041250 IC50 > 30000 nM T23172 C28YFA 127041251 IC50 > 30000 nM T23172 CIP84Z 127041549 IC50 > 30000 nM T23172 CQP76E 127041550 IC50 > 30000 nM T23172 C3A1VL 127041551 IC50 > 30000 nM T23172 CEJ97D 127041858 IC50 = 1130 nM T23172 C35OPG 127041859 IC50 = 2780 nM T23172 CEN15W 127041860 IC50 = 5750 nM T23172 C4UBE5 127041861 IC50 > 30000 nM T23172 C7Q5YC 127045965 IC50 = 39 nM T23172 C3V5BF 127046092 IC50 = 953 nM T23172 C5X2VQ 127046094 IC50 = 716 nM T23172 C2Y1OE 127047142 IC50 = 507 nM T23172 CGA6L4 127047801 IC50 = 584 nM T23172 CB2SE8 127049004 IC50 = 12400 nM T23172 CS6ZO5 127049005 IC50 = 14300 nM T23172 C1PE9L 127050562 IC50 = 1800 nM T23172 CZ5D8C 127050563 IC50 = 20600 nM T23172 CX46RS 127050564 IC50 = 8500 nM T23172 C3LI1J 127050565 IC50 = 1900 nM T23172 CG91WC 127052080 IC50 = 1500 nM T23172 CGQZ74 129048381 IC50 > 10000 nM T23172 C3UH2V 129202507 IC50 = 154 nM T23172 C0XS4M 129896681 IC50 > 10000 nM T23172 CZ13WL 130339268 IC50 > 10000 nM T23172 CXTZ19 131704459 IC50 = 1600 nM T23172 C25WQI 131704460 IC50 = 2 nM T23172 CD4NY1 131839645 IC50 = 397 nM T23172 C6OXE3 132134663 IC50 = 10 nM T23172 CUO0C5 132156633 IC50 > 10000 nM T23172 CV89JM 132231876 IC50 = 41 nM T23172 CK4FI7 132277003 IC50 = 32 nM T23172 C5CZA1 132578411 IC50 = 2440 nM T23172 CH49YN 132962218 IC50 = 7000 nM T23172 CDMF97 134130282 IC50 > 100000 nM T23172 C2H6PW 134130554 IC50 = 4100 nM T23172 CM5T6K 134130825 IC50 = 4800 nM T23172 CWF16B 134131331 IC50 = 7100 nM T23172 CLV5I3 134131586 IC50 = 1800 nM T23172 CC1EB5 134131929 IC50 > 10000 nM T23172 CMZG34 134133313 IC50 = 5970 nM T23172 CX2WN6 134134364 IC50 > 10000 nM T23172 CSZX25 134135323 IC50 = 3490 nM T23172 C56UDO 134135820 IC50 > 100 nM T23172 CA75NE 134135874 IC50 = 183.2 nM T23172 CR6D9H 134136093 IC50 = 836.5 nM T23172 C3G7TQ 134136245 IC50 = 3790 nM T23172 CQH05W 134136683 IC50 = 87.6 nM T23172 C25WAP 134137307 IC50 = 72.6 nM T23172 CQ61HU 134137344 IC50 > 100 nM T23172 CDY10C 134137518 IC50 = 201.8 nM T23172 C6VHL4 134137944 IC50 = 1195.4 nM T23172 CJ7C1N 134137974 IC50 = 793 nM T23172 C4QSZ5 134138566 IC50 > 10000 nM T23172 CZU97C 134138682 IC50 = 6880 nM T23172 C6RGN8 134138812 IC50 > 10000 nM T23172 CA7PD8 134139534 IC50 > 10000 nM T23172 C3OBC6 134139548 IC50 > 10000 nM T23172 CW69GT 134139694 IC50 = 8750 nM T23172 CQE08L 134139702 IC50 = 2420 nM T23172 C8JR1X 134140108 IC50 = 4960 nM T23172 CN1I6V 134140323 IC50 = 70.1 nM T23172 CID3G7 134142328 IC50 = 359.4 nM T23172 C4F6VU 134143525 IC50 = 7670 nM T23172 C41ZEF 134143846 IC50 = 5174 nM T23172 CE43OI 134144225 IC50 = 61.2 nM T23172 CRZ0E5 134146010 IC50 = 7150 nM T23172 CHJ13S 134146699 IC50 = 6940 nM T23172 C3KZV6 134146771 IC50 > 100 nM T23172 C0KNV3 134146887 IC50 = 7620 nM T23172 C4U8KT 134147234 IC50 = 8150 nM T23172 CJ1FQ6 134147869 IC50 = 7440 nM T23172 CXS38A 134147887 IC50 = 7400 nM T23172 C5R2PK 134148588 IC50 > 10000 nM T23172 C0AWH3 134148660 IC50 = 3690 nM T23172 C48AOM 134150297 IC50 = 364.4 nM T23172 CE69LC 134150331 IC50 > 10000 nM T23172 CJ56EZ 134150417 IC50 > 10000 nM T23172 CQK40B 134150618 IC50 > 10000 nM T23172 C10LWI 134151050 IC50 > 100 nM T23172 C43FPY 134151089 IC50 = 67.5 nM T23172 CI4A1T 134152401 IC50 > 10000 nM T23172 C0N6JF 134152887 IC50 = 8010 nM T23172 CG8OY3 134153160 IC50 > 100 nM T23172 C6JFN5 134153988 IC50 = 8880 nM T23172 C4B7IL 134154440 IC50 = 1580.6 nM T23172 C5YX7T 134154596 IC50 > 10000 nM T23172 C07RWN 134154721 IC50 > 10000 nM T23172 CV5M1T 134154754 IC50 = 7100 nM T23172 C9DRQ6 134155700 IC50 = 6450 nM T23172 CUD7A8 134155908 IC50 = 67.2 nM T23172 C6HN5J 134155932 IC50 = 1710 nM T23172 C8CXZ9 134156759 IC50 = 83.1 nM T23172 CQD93J 134156816 IC50 > 10000 nM T23172 C3HCT6 134156845 IC50 = 1220 nM T23172 C3HC0S 134537158 IC50 = 2800 nM T23172 CHK0V4 134611545 IC50 = 96 nM T23172 C20FAE 134611548 IC50 = 92 nM T23172 C51PKU 134611580 IC50 = 98 nM T23172 CJV4Z6 134611726 IC50 = 135 nM T23172 CN75GU 134611727 IC50 = 27 nM T23172 C80PJI 134611728 IC50 = 10 nM T23172 CFM46L 134812674 IC50 > 4950 nM T23172 C2VC5Y 134817793 IC50 > 30000 nM T23172 C54FXD 134957362 IC50 > 10000 nM T23172 CVF86X 135125189 IC50 = 391 nM T23172 C9MCQ0 135138184 IC50 = 1130 nM T23172 C7V2MJ 135142423 IC50 = 56 nM T23172 CLET52 135142442 IC50 = 31 nM T23172 CU13RW 135142625 IC50 = 74 nM T23172 CM7N0J 135142656 IC50 = 221 nM T23172 CG6JI9 135142885 IC50 = 69 nM T23172 CQD32R 135143120 IC50 = 174 nM T23172 CAM74U 135437278 IC50 < 10000 nM T23172 CTJ48K 135524085 IC50 = 1000 nM T23172 CUT1W7 135524168 IC50 = 310 nM T23172 C7PJ6X 135566704 IC50 > 30000 nM T23172 CPHG43 135567142 IC50 = 2.5 nM T23172 C2NRS8 135567293 IC50 = 8.3 nM T23172 C4R1FH 135567294 IC50 = 4.3 nM T23172 CA0R9G 135567295 IC50 = 418.3 nM T23172 CRI5F3 135839295 IC50 = 43.5 nM T23172 CH8W7B 135839328 IC50 = 493.1 nM T23172 C32BOU 135956049 IC50 = 62 nM T23172 CHA4N2 136013680 IC50 > 10 nM T23172 C1YUD0 136219394 IC50 > 10 nM T23172 CIU8W3 136254389 IC50 > 10 nM T23172 C1P6ZW 136263939 IC50 = 1.7 nM T23172 C0R2IL 136901416 IC50 = 3.162 nM T23172 C5JIR2 136987005 IC50 = 78300 nM T23172 CIJ71W 137028350 IC50 = 2400 nM T23172 CS15TL 137028351 IC50 = 2900 nM T23172 CH3M4B 137083628 IC50 > 30000 nM T23172 CJA07O 137083629 IC50 > 30000 nM T23172 C9F8PX 137083630 IC50 > 30000 nM T23172 CE9V4U 137174991 IC50 = 17 nM T23172 CM64UH 137175110 IC50 = 17 nM T23172 C70DIP 137223928 IC50 = 31 nM T23172 C9F3KV 137321155 IC50 = 114.4 nM T23172 CJK67W 137321156 IC50 = 1.65 nM T23172 C3Z4AT 137321159 IC50 = 11 nM T23172 CMY0V2 137321160 IC50 = 0.7 nM T23172 C96CJQ 137348875 IC50 = 3 nM T23172 CWM9S4 137349398 IC50 = 56 nM T23172 C1KSZ6 137475463 IC50 = 2014 nM T23172 C2FT1L 137475480 IC50 = 1033 nM T23172 CAM8K0 137632226 IC50 >= 8000 nM T23172 CH9WK1 137632228 IC50 < 1 nM T23172 C7R2HI 137632648 IC50 >= 8000 nM T23172 C2I3PY 137633211 IC50 = 35 nM T23172 CZH08K 137633516 IC50 = 3 nM T23172 CJN68H 137633647 IC50 >= 8000 nM T23172 CF6RH5 137633780 IC50 = 315 nM T23172 CI1E8V 137634241 IC50 > 10000 nM T23172 COE76K 137634328 IC50 = 2.9 nM T23172 C6IU0M 137634461 IC50 = 656 nM T23172 CE4DH3 137635161 IC50 >= 8000 nM T23172 CXG74K 137635345 IC50 = 5400 nM T23172 C6JVG9 137635398 IC50 = 569 nM T23172 CMV38W 137635509 IC50 = 175 nM T23172 CM73AT 137635759 IC50 >= 8000 nM T23172 CI86AE 137636097 IC50 = 34800 nM T23172 CH5SI7 137636771 IC50 >= 8000 nM T23172 C8I2NQ 137637573 IC50 = 30 nM T23172 C3RF7B 137638414 IC50 >= 8000 nM T23172 CRSE25 137638809 IC50 = 100 nM T23172 CE0ZF8 137638897 IC50 = 1.3 nM T23172 C50WHR 137641404 IC50 >= 8000 nM T23172 CO1MS6 137641896 IC50 = 29000 nM T23172 C2VWE5 137642024 IC50 >= 8000 nM T23172 CJ6PU9 137642141 IC50 = 34.1 nM T23172 C0RX1Z 137642404 IC50 = 556 nM T23172 CA9DE5 137642519 IC50 = 9 nM T23172 C9GDQ6 137642740 IC50 > 1496 nM T23172 C94ELU 137643208 IC50 = 942 nM T23172 CO83EQ 137643608 IC50 = 293.4 nM T23172 CQP79B 137643915 IC50 >= 8000 nM T23172 CGHP09 137645020 IC50 = 0.8 nM T23172 CN34SE 137646319 IC50 = 743 nM T23172 CI8S5A 137646690 IC50 >= 8000 nM T23172 CGE91V 137646834 IC50 >= 8000 nM T23172 CE8SH2 137647292 IC50 = 3.5 nM T23172 CW6D9H 137648009 IC50 >= 8000 nM T23172 CGU2E5 137648767 IC50 = 8 nM T23172 C9KW2L 137648948 IC50 >= 8000 nM T23172 CHN7A3 137648975 IC50 >= 8000 nM T23172 CIB60Q 137649981 IC50 = 1012 nM T23172 CF4X3E 137650150 IC50 > 10000 nM T23172 CVHT54 137650515 IC50 >= 8000 nM T23172 CJQ72A 137650866 IC50 = 372 nM T23172 CA9K6R 137650880 IC50 >= 8000 nM T23172 COCF21 137651256 IC50 = 91 nM T23172 C3Z7LM 137651481 IC50 = 280 nM T23172 CQ27PY 137651710 IC50 = 125 nM T23172 CYA52Z 137652173 IC50 = 783 nM T23172 C5CKI4 137652730 IC50 = 3400 nM T23172 C28QUP 137652864 IC50 = 8160 nM T23172 C6UEB9 137653042 IC50 >= 8000 nM T23172 CK81UT 137654424 IC50 = 1.3 nM T23172 CS6RE8 137654629 IC50 = 8600 nM T23172 CW6SO7 137654686 IC50 >= 8000 nM T23172 CCR5B3 137654793 IC50 = 436 nM T23172 CKM89A 137654900 IC50 = 701 nM T23172 C26ONG 137654955 IC50 >= 8000 nM T23172 CVBS03 137656215 IC50 = 116 nM T23172 CYWE21 137656346 IC50 = 7.1 nM T23172 C6V3WR 137656619 IC50 >= 8000 nM T23172 CT1EP3 137656679 IC50 = 166 nM T23172 CU48SP 137657047 IC50 > 1000 nM T23172 C8VC9A 137657080 IC50 = 16.7 nM T23172 C49DOZ 137657630 IC50 = 3500 nM T23172 C49GYQ 137658008 IC50 >= 8000 nM T23172 C59BVH 137658028 IC50 = 304 nM T23172 CO6C8I 137658504 IC50 >= 8000 nM T23172 CW4CK8 137659037 IC50 > 1496 nM T23172 C6Z8YN 137659188 IC50 = 3600 nM T23172 C86KOS 137659382 IC50 >= 8000 nM T23172 CMZ36T 137659999 IC50 = 1000 nM T23172 CR41KW 137660124 IC50 = 196 nM T23172 CQ8KF2 137660642 IC50 >= 8000 nM T23172 COMQ54 137661391 IC50 >= 8000 nM T23172 CJ52WM 137661888 IC50 >= 8000 nM T23172 CU2L5H 138108525 EC50 = 237 nM T23172 C2W0JU 138319690 IC50 > 30000 nM T23172 CXV84M 138377596 IC50 = 7.4 nM T23172 C8X9DR 138584993 IC50 = 75.03 nM T23172 C9NL1M 138585023 IC50 = 1.09 nM T23172 CHX6N7 138585027 IC50 = 2.55 nM T23172 C3RM2Z 138585033 IC50 = 2.92 nM T23172 CBF8S4 138585069 IC50 = 818.9 nM T23172 C4O0GC 138585070 IC50 = 6.65 nM T23172 C7KYU3 138585074 IC50 = 87.03 nM T23172 CE5S4Z 138585101 IC50 = 1111.5 nM T23172 CM63FA 138585111 IC50 = 18.31 nM T23172 C2U8PZ 138585129 IC50 = 27.5 nM T23172 C0Y2WZ 138585150 IC50 = 129.75 nM T23172 CHMX08 138585151 IC50 = 1.01 nM T23172 CA8N5T 138585156 IC50 = 124.1 nM T23172 CG8TR3 138585164 IC50 = 23.45 nM T23172 C3JR7K 138585184 IC50 = 26.58 nM T23172 CQI78V 138585192 IC50 = 143.7 nM T23172 C2UCN9 138605457 IC50 = 9.94 nM T23172 C3RM1U 138605458 IC50 = 285.9 nM T23172 CD4M3W 138605461 IC50 = 28.94 nM T23172 C4VMQ9 138605557 IC50 = 95.56 nM T23172 CQ6R7X 138911330 IC50 > 10000 nM T23172 CI1D9F 139600335 IC50 = 39 nM T23172 C9ZYG8 141366083 IC50 = 15000 nM T23172 C18QDP 141523774 IC50 = 20.7 nM T23172 CD9F4Y 141523776 IC50 = 34 nM T23172 C4L6JD 141523781 IC50 = 41.1 nM T23172 CLOI54 141523782 IC50 = 932.9 nM T23172 CDF78Y 141523783 IC50 = 397 nM T23172 CSZQ36 141523784 IC50 = 80.5 nM T23172 CTYQ49 141523785 IC50 = 103.2 nM T23172 C8FC9Y 141531439 IC50 = 197.2 nM T23172 CU51PI 141531440 IC50 = 9.9 nM T23172 C81RPA 141531442 IC50 = 19.2 nM T23172 CAT46B 141531443 IC50 = 6.2 nM T23172 CS37YV 141531444 IC50 = 582.6 nM T23172 CN75MA 141728817 IC50 = 7.6 nM T23172 C7EL5X 141728840 IC50 = 2 nM T23172 C9H8PX 141728841 IC50 = 3.3 nM T23172 CC03XH 141728860 IC50 = 3.7 nM T23172 CECS13 141753441 IC50 = 2.4 nM T23172 C1JR5B 142379949 IC50 = 106 nM T23172 C47YDW 142744361 IC50 = 1760 nM T23172 C2OA9H 145949725 IC50 = 464 nM T23172 CY04PB 145950223 IC50 = 18100 nM T23172 CDTW63 145950378 IC50 > 30000 nM T23172 CDJ81U 145952312 IC50 > 30000 nM T23172 C2XP8N 145953005 IC50 > 30000 nM T23172 CN0V3D 145953512 IC50 > 30000 nM T23172 C1OQ3J 145953599 IC50 > 27900 nM T23172 CNS52L 145954024 IC50 > 30000 nM T23172 CRU9F8 145955362 IC50 > 30000 nM T23172 CIP2J9 145955397 IC50 = 20300 nM T23172 CQ68WS 145956107 IC50 = 371 nM T23172 CZ0B7A 145956262 IC50 > 30000 nM T23172 CO6SV3 145957001 IC50 > 30000 nM T23172 C51ADW 145958260 IC50 = 24600 nM T23172 C3L8IE 145958641 IC50 = 517 nM T23172 C7B2LD 145959014 IC50 = 12600 nM T23172 CO05IK 145959360 IC50 = 144 nM T23172 CMCG17 145959462 IC50 = 6540 nM T23172 CEN74X 145960527 IC50 = 205 nM T23172 C2LD5V 145960573 IC50 > 30000 nM T23172 CN02MC 145961070 IC50 = 11 nM T23172 CQ1G2E 145961384 IC50 = 505 nM T23172 CUG21K 145961523 IC50 > 1000 nM T23172 CFY21D 145961655 IC50 = 0.39 nM T23172 CN6T7U 145961668 IC50 = 59 nM T23172 CL9U6P 145961765 IC50 = 436 nM T23172 C5YP6V 145962131 IC50 = 30 nM T23172 C49SBC 145962154 IC50 = 642 nM T23172 CK27PU 145962349 IC50 = 390 nM T23172 CKYH98 145962459 IC50 = 678 nM T23172 CSF4Y9 145962642 IC50 = 368 nM T23172 CUVF80 145962646 IC50 = 129 nM T23172 CI9Z7U 145962747 IC50 = 48 nM T23172 CW8S0D 145962858 IC50 = 571 nM T23172 CJ4D3N 145963061 IC50 = 490 nM T23172 C1O6TU 145963095 IC50 > 10000 nM T23172 CQXL78 145963239 IC50 = 23 nM T23172 CQ86LZ 145963345 EC50 = 257 nM T23172 C9ZJ7H 145963618 IC50 = 499 nM T23172 CEDZ18 145971190 IC50 > 30000 nM T23172 CKPM09 145971514 IC50 > 30000 nM T23172 C7K1AJ 145971681 IC50 = 121 nM T23172 C7OD0E 145973587 IC50 = 18100 nM T23172 CE36NY 145979199 IC50 > 100 nM T23172 CHVD06 145979212 IC50 = 0.5 nM T23172 C7L1IC 145979240 IC50 = 38 nM T23172 CAJ37B 145979552 IC50 = 13 nM T23172 CXE8H0 145979687 IC50 = 11.23 nM T23172 CE31VG 145979714 IC50 = 3 nM T23172 C7N8DU 145980127 IC50 = 230 nM T23172 CA2CD1 145980524 IC50 > 100 nM T23172 C8AMK1 145980722 IC50 = 6 nM T23172 C81XFH 145980840 IC50 = 2 nM T23172 CR43KU 145980943 IC50 = 21.59 nM T23172 C85XBC 145981348 IC50 = 26 nM T23172 C6M1CP 145981406 IC50 > 100 nM T23172 CCR27P 145982758 IC50 = 787.5 nM T23172 CMWO35 145982855 IC50 > 1000 nM T23172 CEU47V 145983063 IC50 = 189.3 nM T23172 C5VF8P 145983087 IC50 = 15.6 nM T23172 C35FMR 145983116 IC50 > 500 nM T23172 C0YFS6 145983170 IC50 > 500 nM T23172 CWS14X 145983289 IC50 = 143.2 nM T23172 CV28DA 145983327 IC50 = 373.7 nM T23172 C57KUM 145983360 IC50 > 1000 nM T23172 CF41KU 145983453 IC50 = 315.3 nM T23172 CS1GK8 145983460 IC50 = 56.1 nM T23172 C48ZXP 145983545 IC50 = 196 nM T23172 CG97VS 145983548 IC50 = 87.4 nM T23172 CML89J 145983552 IC50 = 144.2 nM T23172 C9UJR1 145983646 IC50 > 1000 nM T23172 CA20KM 145983867 IC50 = 21.3 nM T23172 CS58RN 145983989 IC50 = 115.4 nM T23172 C7D8IA 145983997 IC50 > 1000 nM T23172 CM8Z7V 145984082 IC50 = 496 nM T23172 CXMO36 145984108 IC50 = 278.4 nM T23172 C7THN1 145984160 IC50 = 66 nM T23172 C30EHD 145984172 IC50 = 16 nM T23172 CN0GU3 145984181 IC50 > 1000 nM T23172 C8CQK3 145984479 IC50 = 267.4 nM T23172 CP8J3H 145984569 IC50 = 124.4 nM T23172 C42SJR 145984669 IC50 = 57.7 nM T23172 CLH7K9 145984673 IC50 = 94.3 nM T23172 C67HUC 145984822 IC50 = 32.3 nM T23172 C0PT2V 145984960 IC50 = 154.2 nM T23172 CW7H0X 145984995 IC50 = 756.3 nM T23172 CG4U3I 145985120 IC50 = 36.3 nM T23172 CD1T8G 145985288 IC50 > 1000 nM T23172 C3U9IS 145985565 IC50 = 324.3 nM T23172 CXQ2O9 145985661 IC50 > 100 nM T23172 C2HXR3 145985769 IC50 = 394.8 nM T23172 CY7X5L 145986106 IC50 = 591.2 nM T23172 C17TBU 145986946 IC50 = 6.77 nM T23172 C2JCA0 145987101 IC50 = 120 nM T23172 CNV15E 145987655 IC50 > 100 nM T23172 C52AOJ 145987765 IC50 = 1.39 nM T23172 C8NEY2 145987871 IC50 = 0.9 nM T23172 CHAE74 145987939 IC50 > 100 nM T23172 C9KJ1A 145988137 IC50 = 1 nM T23172 C9BX4U 145988956 IC50 = 0.5 nM T23172 CPH14J 145989239 IC50 > 100 nM T23172 CIVK73 145989244 IC50 = 1 nM T23172 CL1IV0 145989334 IC50 = 0.83 nM T23172 CGB2F6 145989547 IC50 = 0.95 nM T23172 CC8GZ3 145989610 IC50 = 6 nM T23172 C5I8SR 145989639 IC50 = 1226 nM T23172 C82FRH 145989705 IC50 = 0.69 nM T23172 CLM9U8 145989960 IC50 > 100 nM T23172 CIU9W4 145990027 IC50 = 5828 nM T23172 CQH40O 145990342 IC50 = 1.06 nM T23172 C3DWZ0 145990496 IC50 = 953 nM T23172 CTX1A3 145990814 IC50 = 7 nM T23172 C6LSR8 145990895 IC50 = 8.34 nM T23172 CNG35K 145991262 IC50 = 12 nM T23172 C0M6LD 145991292 IC50 = 14 nM T23172 CKGE38 145991618 IC50 = 7 nM T23172 C71HFI 145992300 IC50 = 91.15 nM T23172 CI8R6P 145992803 IC50 = 3 nM T23172 CP7KE0 145992836 IC50 > 100 nM T23172 CD09RT 145992905 IC50 = 80.1 nM T23172 CR2F1Y 145993348 IC50 = 13 nM T23172 C51DMH 145993445 IC50 = 1 nM T23172 CR5OL0 145993847 IC50 > 100 nM T23172 CYZ72C 145994233 IC50 = 0.91 nM T23172 CHQU21 146185142 IC50 = 1759 nM T23172 C71KXB 146185156 IC50 = 965 nM T23172 C9IA1X 146185163 IC50 = 1584 nM T23172 CS0OL6 146185170 IC50 = 513 nM T23172 C1IAH7 146185174 IC50 = 2788 nM T23172 C8JWQ5 146266924 IC50 = 1777 nM T23172 C4V2IZ 146266925 IC50 = 0.4 nM T23172 C43FOQ 147462647 IC50 > 1000 nM T23172 C5DAO2 149003255 IC50 > 1000 nM T23172 CXY6S2 150234011 IC50 = 52 nM T23172 CP0B5C 150773469 Ki = 1 nM T23172 CK0H4X 150894694 IC50 = 817 nM T23172 C7PLT9 155510967 IC50 > 10000 nM T23172 C1WRE2 155511764 IC50 = 39 nM T23172 CR1SE8 155511850 IC50 = 8737 nM T23172 C91YXU 155511860 IC50 = 873.2 nM T23172 CDY5U0 155512704 IC50 = 109.4 nM T23172 CT9B4M 155512787 IC50 = 741.3 nM T23172 C2MD1Q 155513187 IC50 > 10000 nM T23172 CM95KR 155513637 IC50 = 335.7 nM T23172 C59BGM 155514196 IC50 = 19 nM T23172 C83ZSG 155514311 IC50 = 4 nM T23172 C7MJY5 155514805 IC50 = 2 nM T23172 C7AMX8 155514903 IC50 = 84 nM T23172 CQH6P0 155514988 IC50 = 5.4 nM T23172 CUIO35 155516044 IC50 = 98.1 nM T23172 CD6YR0 155516192 IC50 = 267.4 nM T23172 CI23DH 155516489 IC50 = 123 nM T23172 CTP29J 155516678 IC50 = 1.4 nM T23172 CYH8Z6 155517558 IC50 = 21 nM T23172 C57JLV 155517837 IC50 = 21 nM T23172 C0E7WS 155518120 IC50 = 4962 nM T23172 CDTG10 155518349 IC50 < 1 nM T23172 C3NA2I 155519537 IC50 > 1000 nM T23172 CF0H9V 155520176 IC50 > 3000 nM T23172 C0A9LX 155520276 IC50 > 10000 nM T23172 C4YJN9 155520341 IC50 = 6494 nM T23172 C0YEX7 155521332 IC50 = 13 nM T23172 CLZ08K 155522634 IC50 = 783.9 nM T23172 CXG4L3 155522806 IC50 = 3.5 nM T23172 CEU10G 155522970 IC50 = 751 nM T23172 C7NVQ5 155523535 IC50 = 240.1 nM T23172 C32POG 155523862 IC50 = 683 nM T23172 CSVH92 155523915 IC50 = 0.6 nM T23172 C1HWG6 155524274 IC50 > 1000 nM T23172 CHO23V 155525901 IC50 = 4000 nM T23172 CE4FX7 155525956 IC50 = 364.1 nM T23172 C39EGQ 155526165 IC50 = 689.2 nM T23172 CRT67D 155526236 IC50 = 1.2 nM T23172 CE3OH1 155527121 IC50 = 11 nM T23172 CI80JY 155527297 IC50 = 7.5 nM T23172 CCS24O 155527492 IC50 = 89.6 nM T23172 CK14UT 155528172 IC50 > 10000 nM T23172 CB26JT 155528364 IC50 = 8 nM T23172 CU1HB3 155528554 IC50 = 894 nM T23172 C4V3EX 155528562 IC50 = 16 nM T23172 C1VE9C 155528748 IC50 = 2 nM T23172 CVW07K 155528897 IC50 = 103 nM T23172 CMIC15 155529301 IC50 = 552.4 nM T23172 CAZ3N2 155529440 IC50 = 21 nM T23172 CL47NH 155529550 IC50 = 160 nM T23172 C5QRB3 155529779 IC50 = 0.4 nM T23172 CUXA18 155529935 IC50 = 51 nM T23172 CF7HU2 155530436 IC50 = 4.4 nM T23172 CL0US4 155530459 IC50 = 0.6 nM T23172 CX0B9Q 155530477 IC50 = 111.8 nM T23172 CU34BK 155530609 IC50 = 0.4 nM T23172 C2WCU6 155530774 IC50 = 470 nM T23172 C67TQL 155530972 IC50 = 481.7 nM T23172 C4LE7Q 155532724 IC50 = 3 nM T23172 CLSV71 155533995 IC50 = 180 nM T23172 C1NGV5 155534208 IC50 = 24 nM T23172 C51ZMX 155534302 Ki = 3.3 nM T23172 CGH63O 155534464 IC50 = 1 nM T23172 C2NPE6 155534808 IC50 = 11 nM T23172 C64FIW 155534972 IC50 > 10000 nM T23172 CE8QW2 155535975 IC50 = 5 nM T23172 CQIB17 155536661 IC50 < 0.1 nM T23172 C2CG1A 155537016 IC50 > 10000 nM T23172 C06JDH 155537151 IC50 = 18 nM T23172 C5GNH8 155538704 IC50 > 3000 nM T23172 CGV96F 155538868 IC50 = 41 nM T23172 C3O6KI 155540160 IC50 > 3000 nM T23172 C0D8OL 155540191 IC50 = 10 nM T23172 CP2NY0 155540484 IC50 = 2.512 nM T23172 CF8O5T 155540488 IC50 = 1000 nM T23172 C51JNT 155540621 IC50 = 3.162 nM T23172 C5BTX7 155540994 IC50 > 1000 nM T23172 CT1AX5 155541077 IC50 = 2.512 nM T23172 CY8F7S 155541097 IC50 > 10000 nM T23172 CH6LV1 155541475 IC50 = 12.59 nM T23172 CS58BA 155541478 IC50 = 4.84 nM T23172 CXM43A 155542056 IC50 = 21 nM T23172 CH10DU 155542091 IC50 = 104 nM T23172 CF9AX3 155542099 IC50 = 16 nM T23172 CO82TS 155542339 IC50 = 290 nM T23172 C1B6EK 155542401 IC50 = 3.981 nM T23172 CH59RW 155542578 IC50 = 2477 nM T23172 C23PZE 155542904 IC50 = 4 nM T23172 CKL31P 155542961 IC50 = 25.12 nM T23172 CH46TG 155543289 IC50 = 24.1 nM T23172 C1QRZ2 155543349 IC50 = 6872 nM T23172 CW73EO 155543439 IC50 = 4.2 nM T23172 CKM8G4 155543489 IC50 = 89 nM T23172 CRA21U 155543538 IC50 = 8.4 nM T23172 CD9Z3W 155544141 IC50 = 1.1 nM T23172 CWSG67 155544202 IC50 = 837 nM T23172 C4PO7Q 155544443 IC50 = 278 nM T23172 CTQ63L 155544706 IC50 = 12.59 nM T23172 CP7XE1 155545114 IC50 = 1.995 nM T23172 CFR42U 155545338 IC50 = 31.62 nM T23172 C5U8HP 155546232 IC50 = 7.943 nM T23172 CBK0O4 155547208 IC50 = 6.4 nM T23172 CSI1U9 155547916 IC50 = 2531 nM T23172 C0B3RK 155547921 IC50 = 63.1 nM T23172 C67AYP 155548399 IC50 = 430.7 nM T23172 C63EKL 155548728 IC50 = 873 nM T23172 CT5EM7 155548782 IC50 = 212 nM T23172 CI6Y5Z 155549690 IC50 = 2.512 nM T23172 C10OSG 155550219 IC50 = 15 nM T23172 C3DW8J 155550308 IC50 = 3.981 nM T23172 C31QUW 155550462 IC50 = 1 nM T23172 C6UJS7 155550600 IC50 = 38 nM T23172 CAZ51Y 155551384 IC50 = 6 nM T23172 C0DMP2 155551420 IC50 = 9.4 nM T23172 CE73NZ 155552094 Ki = 55 nM T23172 CX0HL6 155552133 IC50 = 603.2 nM T23172 CW1UX0 155552333 IC50 = 6.31 nM T23172 C0HUL3 155552710 IC50 = 3.7 nM T23172 C62ERW 155552853 IC50 = 31.62 nM T23172 CI2BZ9 155553084 IC50 = 104 nM T23172 CPB6M8 155553409 IC50 = 3.5 nM T23172 C5HQ7X 155553551 IC50 = 2 nM T23172 CNTP52 155554413 IC50 = 3078 nM T23172 CWLC85 155554605 IC50 = 171.8 nM T23172 C2GB5O 155554793 IC50 = 232 nM T23172 CQ6S8E 155554939 IC50 = 7.943 nM T23172 CP39ZD 155555305 IC50 = 63.1 nM T23172 C9J4HM 155555486 IC50 > 10000 nM T23172 C6TPL9 155556222 IC50 = 27 nM T23172 C2VS8X 155556321 IC50 = 342 nM T23172 CG48UE 155556474 IC50 = 3.162 nM T23172 C8TYG7 155556520 IC50 > 10000 nM T23172 C59HKP 155557055 IC50 = 589 nM T23172 CH9ON1 155557340 IC50 = 155 nM T23172 CHW4O3 155558352 IC50 = 3.162 nM T23172 C7HFI8 155558403 IC50 = 23 nM T23172 C2LK9V 155558426 IC50 = 99 nM T23172 C7WND0 155558729 IC50 > 10000 nM T23172 CPAV79 155559005 IC50 = 61 nM T23172 C3V5HL 155559143 IC50 = 70.4 nM T23172 C2U5ZM 155559343 IC50 = 5.012 nM T23172 CSF54R 155559609 IC50 = 7.3 nM T23172 CANJ25 155559746 IC50 = 251.19 nM T23172 C46KLS 155559780 IC50 = 260.1 nM T23172 C51IBQ 155560019 IC50 = 186 nM T23172 CNK81M 155560413 IC50 = 25.12 nM T23172 C54NQC 155561203 IC50 = 2878 nM T23172 C1Z6IL 155561218 IC50 > 3000 nM T23172 CH1LJ2 155562424 IC50 = 389 nM T23172 C68TCL 155563799 IC50 = 7 nM T23172 CAC85T 155564156 IC50 = 1428 nM T23172 CBQN81 155564466 IC50 = 7.2 nM T23172 CY9VK1 155564952 IC50 = 0.6 nM T23172 CZ2NK9 155565077 IC50 = 2511.89 nM T23172 CM02CX 155565267 IC50 > 1000 nM T23172 CSNF76 155565806 IC50 = 3.981 nM T23172 CF1X5I 155566525 IC50 > 10000 nM T23172 C7S5MC 155566661 IC50 = 730 nM T23172 C6AXL1 155567447 IC50 = 101 nM T23172 CSRZ04 155567801 IC50 > 3000 nM T23172 COS7X5 155568028 IC50 = 245.2 nM T23172 COGC41 155568181 IC50 = 319.3 nM T23172 C0L6UT 155568261 IC50 = 15.85 nM T23172 CR79DJ 155568314 IC50 > 3000 nM T23172 C8EYW3 155568955 IC50 = 9.3 nM T23172 CGU74Q 155569301 IC50 = 69 nM T23172 C6JKT9 16750206 IC50 > 10000 nM T23172 CYIU14 16750228 IC50 = 620 nM T23172 COM3C1 16750290 IC50 = 720 nM T23172 CI67WG 16750292 IC50 = 89 nM T23172 CL2SY5 16750330 IC50 = 7200 nM T23172 CE5P2I 53363072 IC50 = 1600 nM T23172 CTV60O 53363073 IC50 = 2500 nM T23172 CD74BW 53363074 IC50 = 6000 nM T23172 CU3M8P 53363075 IC50 > 10000 nM T23172 C07FTA 53363076 IC50 > 10000 nM T23172 C9JX2G 53363150 IC50 = 750 nM T23172 CJ04SF 53363151 IC50 = 500 nM T23172 CO7Z2P 53363152 IC50 = 380 nM T23172 C1T2LY 53363154 IC50 = 830 nM T23172 C9GEA7 53363242 IC50 = 3300 nM T23172 CTSP38 53363245 IC50 = 390 nM T23172 CM7BZ3 53363246 IC50 = 1000 nM T23172 CU76JB 53363338 IC50 = 890 nM T23172 C2PU3M 53364335 IC50 > 10000 nM T23172 C10FXI 53364337 IC50 = 1200 nM T23172 C2U9QE 53364338 IC50 = 1100 nM T23172 D00ATA 5908088 IC50 = 900 nM T23172 D00ERW 44444843 Ki > 1722 nM T23172 D00HVA 11624601 Ki > 1700 nM T23172 D01RHR 71519693 IC50 = 1705 nM T23172 D01VFR 4708 IC50 = 3140 nM T23172 D02BXJ 46864270 IC50 = 57.5 nM T23172 D02NNT 53232451 IC50 = 7 nM T23172 D02PVB 8515 IC50 = 957 nM T23172 D03BQI 3794 IC50 = 9100 nM T23172 D05MHL 44605611 Ki = 0.0055 nM T23172 D06BJG 71556703 IC50 = 6370 nM T23172 D06HVH 54613583 IC50 > 10000 nM T23172 D06LJL 9916282 IC50 = 25000 nM T23172 D06WGX 9549184 IC50 > 25000 nM T23172 D07OXC 11650194 IC50 > 8300 nM T23172 D08HFG 24809764 IC50 > 10000 nM T23172 D08RZB 11153014 IC50 = 6 nM T23172 D09HVH 135566652 IC50 > 10 nM T23172 D09HXU 16086113 IC50 = 9819 nM T23172 D0E5IP 3795 IC50 = 1800 nM T23172 D0GN5Z 5281295 IC50 = 4260 nM T23172 D0H7DQ 6419755 IC50 = 17 nM T23172 D0IR6U 5494425 IC50 = 5 nM T23172 D0J3LR 11634725 Ki > 4000 nM T23172 D0O6OH 71553154 IC50 = 5300 nM T23172 D0OP3D 25099184 IC50 = 9 nM T23172 D0OZ2S 11785878 IC50 = 150 nM T23172 D0Q3NG 11715520 Ki > 1700 nM T23172 D0S7IE 11658882 Ki > 1700 nM T23172 D0US9O 45275255 IC50 = 35 nM T23172 D0V6VQ 53344620 IC50 = 139.3 nM T23172 D0VC0I 5169 IC50 > 100000 nM T23172 D0YX5U 3797 IC50 = 80 nM T23172 D0Z7TM 22273644 IC50 > 50000 nM T01037 D0I9JH 122070 IC50 = 2600 nM T01037 D0K2ER 3651377 IC50 = 1600 nM T01037 C2XQI7 11526708 IC50 = 3 nM T01037 C45NBF 11705274 IC50 > 30000 nM T01037 CK3Z7D 14591236 IC50 = 3200 nM T01037 C1WJ2D 16070041 IC50 > 30000 nM T01037 C47QOB 19914713 IC50 > 10000 nM T01037 CXV9I2 44389535 IC50 > 10000 nM T01037 C9O7QC 44389542 IC50 = 6700 nM T01037 CK67MQ 44389574 IC50 = 7200 nM T01037 CH2V4K 44389592 IC50 = 3200 nM T01037 CDF0C1 44389649 IC50 > 10000 nM T01037 CZ4P1W 44389720 IC50 = 900 nM T01037 C7RO8N 44389925 IC50 = 6400 nM T01037 CF6HQ0 44389930 IC50 = 290 nM T01037 CX19CD 44389950 IC50 = 650 nM T01037 C2WIP5 44390020 IC50 = 260 nM T01037 CUW8S1 44390083 IC50 = 250 nM T01037 CG26JE 44390119 IC50 = 1100 nM T01037 C5W9NV 44390220 IC50 = 4300 nM T01037 CH90OQ 44390282 IC50 = 330 nM T01037 CI3F2O 44390366 IC50 = 600 nM T01037 CWN08I 44390496 IC50 = 22 nM T01037 CIHV20 44390555 IC50 = 160 nM T01037 C6XN8F 44390610 IC50 = 16 nM T01037 C1K5JB 44390653 IC50 = 5 nM T01037 CI3BM4 44390722 IC50 = 7 nM T01037 C3F6XS 44390723 IC50 = 32 nM T01037 CUJG39 44390835 IC50 = 12 nM T01037 CXW9Z3 44390875 IC50 = 8 nM T01037 C69GNE 44390943 IC50 = 4 nM T01037 CED76T 44390981 IC50 = 6 nM T01037 C8GXP9 44391207 IC50 = 33 nM T01037 C7SO2E 44391283 IC50 = 31 nM T01037 C4MH8K 51355427 IC50 = 3200 nM T01037 CNJ4A8 51355697 IC50 > 30000 nM T01037 CWZ94B 51355698 IC50 > 30000 nM T01037 CM2SH9 51355699 IC50 > 30000 nM T01037 C6CEN7 51355700 IC50 > 30000 nM T01037 CG4L0N 51355701 IC50 > 30000 nM T01037 C6T1IN 51355702 IC50 > 30000 nM T01037 C0X3DU 51355965 IC50 > 30000 nM T01037 CEXJ19 51355966 IC50 > 30000 nM T01037 C2XGZ3 51355967 IC50 > 30000 nM T01037 CYE47P 51355968 IC50 > 30000 nM T01037 CSK29T 51355969 IC50 > 30000 nM T01037 CS9V6B 51356246 IC50 > 30000 nM T01037 C04TKO 51356247 IC50 > 30000 nM T01037 CP7Q0N 53316966 IC50 > 30000 nM T01037 D0W6TB 16730275 IC50 > 30000 nM T86273 D03ZTE 10133 EC50 = 6100 nM T86273 D04DJN 10635 EC50 = 4490 nM T86273 D06XMU 6013 EC50 = 18300 nM T86273 D07BSQ 5994 EC50 = 2770 nM T86273 D08QMX 5757 EC50 = 38400 nM T86273 D0D1SG 5755 IC50 = 251 nM T86273 D0G3SH 31401 EC50 = 2390 nM T86273 D0K0EK 5881 EC50 = 3330 nM T86273 D0M4WA 447715 EC50 = 100 nM T86273 D0OR2L 221493 EC50 = 13600 nM T86273 D02PQB 222528 EC50 = 1250 nM T86273 D04SLF 9903 EC50 = 580 nM T86273 D09NTG 6675 EC50 = 4950 nM T86273 D0H5HO 5879 EC50 = 6220 nM T86273 D0O8FW 441302 EC50 = 3200 nM T86273 D0R9YR 64971 EC50 = 1040 nM T86273 CPV01Q 15818 EC50 = 7010 nM T86273 C91OFE 64980 EC50 = 3110 nM T86273 CKH0W1 73170 EC50 > 10000 nM T86273 CLM3Y7 73493 EC50 > 10000 nM T86273 CQT19P 73641 EC50 > 10000 nM T86273 CO7E1J 91472 EC50 > 10000 nM T86273 CC1LA4 92158 EC50 > 10000 nM T86273 C19WAN 92803 EC50 = 6080 nM T86273 C9A1UP 92810 EC50 = 290 nM T86273 CPBA32 92880 EC50 = 590 nM T86273 CRP79K 94192 EC50 = 10930 nM T86273 C61KXR 114611 EC50 = 36700 nM T86273 CXQ5O3 115245 EC50 = 540 nM T86273 C2EWK9 119046 EC50 = 24200 nM T86273 CR3C1L 122844 EC50 = 4710 nM T86273 CY6G0E 126016 EC50 = 76 nM T86273 CL0VY3 134494 EC50 = 2440 nM T86273 CRL43B 192254 EC50 = 47200 nM T86273 COW8H3 219833 EC50 = 850 nM T86273 CNYA81 247732 EC50 = 2620 nM T86273 CR4HK3 440071 EC50 = 47800 nM T86273 CEX6R9 447718 EC50 = 14500 nM T86273 CC4X3R 451489 EC50 > 100000 nM T86273 CWO27K 463452 EC50 > 10000 nM T86273 C1UQ6Y 723048 EC50 = 3162.28 nM T86273 CI5JS2 749179 EC50 = 3981.07 nM T86273 CLQ8H5 1434463 EC50 = 1310 nM T86273 CFV8I5 1452520 EC50 = 350 nM T86273 CR5QV4 1452523 EC50 > 80000 nM T86273 C45MBQ 1452577 EC50 = 5800 nM T86273 C6XO8U 2733768 EC50 = 680 nM T86273 CT34VY 3223370 EC50 = 880 nM T86273 C9G8HR 5283820 EC50 = 31600 nM T86273 C26NCP 5283821 EC50 = 4890 nM T86273 C6EYM9 5283932 EC50 = 3980 nM T86273 C3H8WR 5284055 EC50 = 870 nM T86273 C09QOX 5284060 EC50 = 120 nM T86273 C4EV1S 5284061 EC50 = 2180 nM T86273 C04TGD 5284305 EC50 = 24400 nM T86273 CEM24L 7203539 EC50 > 102000 nM T86273 C7BEU4 9910920 EC50 = 4790 nM T86273 CW34HS 9929677 EC50 = 10400 nM T86273 C8TC9O 10161414 EC50 > 10000 nM T86273 CDR7X8 10415328 EC50 > 10000 nM T86273 CI1G2S 10479586 EC50 = 5020 nM T86273 CL4UF8 10838116 EC50 > 10000 nM T86273 CKG6N5 11069533 EC50 = 4390 nM T86273 CB03TK 11143041 EC50 > 316000 nM T86273 CSM3P4 11165617 EC50 = 1330 nM T86273 CRHE62 11258221 EC50 = 75700 nM T86273 C7LD6U 11281160 EC50 > 100000 nM T86273 C9PI2O 11281589 EC50 = 1490 nM T86273 C6YD9N 11463847 EC50 = 2910 nM T86273 C4N9EJ 11656002 EC50 = 0.23 nM T86273 CN76YO 12113821 EC50 = 5000 nM T86273 CWA8J6 17755103 EC50 = 2830 nM T86273 CW8OL6 17755104 IC50 = 140 nM T86273 C35DEL 21121407 EC50 = 440 nM T86273 CC8JB3 24721570 EC50 > 10000 nM T86273 C2O3WR 24969527 IC50 = 65 nM T86273 C91HRW 24969872 EC50 = 154 nM T86273 C4BCY2 24969952 IC50 = 44 nM T86273 C2K6WY 26404327 IC50 = 97 nM T86273 CF39AZ 42429922 IC50 = 580 nM T86273 CKD2B8 44337790 EC50 = 2170 nM T86273 CY5R4B 44372731 EC50 = 770 nM T86273 CU9N8E 44372853 EC50 = 1250 nM T86273 C2K6ZW 44427760 EC50 = 3580 nM T86273 C8TYE6 44427761 EC50 = 140 nM T86273 CI86EY 44427762 EC50 = 95 nM T86273 C9U3OY 44427763 EC50 = 4390 nM T86273 C5K7DN 44427764 EC50 = 25500 nM T86273 CS0Y9I 44427765 EC50 > 51900 nM T86273 C9XQO6 44457460 EC50 = 2290 nM T86273 CBKD67 44457463 EC50 > 100000 nM T86273 CM02GU 44457471 EC50 = 250 nM T86273 C6LFG1 44457475 EC50 = 360 nM T86273 C20TGE 44457480 EC50 = 730 nM T86273 CYQM83 44457490 EC50 = 1000 nM T86273 CQ21YX 44457491 EC50 = 2360 nM T86273 C2OI7T 44457500 EC50 = 780 nM T86273 CK80JN 44457504 EC50 = 2630 nM T86273 C9QN7Z 44457506 EC50 = 6180 nM T86273 CY8G7E 44479724 EC50 = 6910 nM T86273 C2YX6O 44605418 EC50 = 820 nM T86273 C8P3NE 44605615 EC50 = 5011.87 nM T86273 C89VRG 44605616 EC50 = 31.62 nM T86273 CZD25I 44605617 EC50 = 23 nM T86273 CT02KM 44626488 EC50 > 10000 nM T86273 COR8X5 44626598 EC50 > 10000 nM T86273 CT3L9B 44626599 EC50 = 3170 nM T86273 C8PS2J 44626600 EC50 = 7880 nM T86273 C36EYX 44626704 EC50 = 7730 nM T86273 C3QMF6 44626706 EC50 > 10000 nM T86273 C6QL2K 44626707 EC50 > 10000 nM T86273 CY5J3Z 44626807 EC50 > 10000 nM T86273 C4AJ7S 44626808 EC50 > 10000 nM T86273 CFH7J6 44626897 EC50 > 10000 nM T86273 CP58DB 44626898 EC50 > 10000 nM T86273 C9REG8 44626899 EC50 > 10000 nM T86273 C32OBM 44626900 EC50 > 10000 nM T86273 C2FV4B 44626993 EC50 > 10000 nM T86273 CHQN53 44626994 EC50 > 10000 nM T86273 CUC03X 44626996 EC50 > 10000 nM T86273 C6L7EJ 44627091 EC50 > 10000 nM T86273 C39HRT 44627092 EC50 > 10000 nM T86273 C61DAY 44627094 EC50 > 10000 nM T86273 CUS18N 44627197 EC50 > 10000 nM T86273 C7JFV4 44627198 EC50 > 10000 nM T86273 CWNU96 44627199 EC50 > 10000 nM T86273 C5VOB1 44627200 EC50 > 10000 nM T86273 CT2CJ8 44627310 EC50 = 3320 nM T86273 C8V2TL 44627311 EC50 = 2080 nM T86273 CS3AU5 44627312 EC50 = 120 nM T86273 CL0OX4 44627313 EC50 = 6270 nM T86273 CQH95P 44627314 EC50 = 420 nM T86273 C9XD1O 45273910 EC50 = 6.1 nM T86273 C1GZV8 45483944 EC50 = 95 nM T86273 CZAC04 45485269 EC50 > 10000 nM T86273 C4O5VH 45485277 EC50 = 3650 nM T86273 C60GHQ 45485278 EC50 > 10000 nM T86273 C1PZ7D 45485281 EC50 > 10000 nM T86273 CU3T9P 45485282 EC50 > 10000 nM T86273 CB1I6M 46195848 EC50 = 10 nM T86273 CX6QC1 46232359 EC50 = 2511.89 nM T86273 CRO8V7 46232360 EC50 = 12.59 nM T86273 C42GBO 46232361 EC50 = 19.95 nM T86273 CO27DY 46232410 EC50 = 1000 nM T86273 CNU72W 46232411 EC50 = 6309.57 nM T86273 C6TR4S 46232412 EC50 = 1258.93 nM T86273 C5Z6HD 46232413 EC50 = 7943.28 nM T86273 C5K0CT 46232414 EC50 = 19.95 nM T86273 C5RX3N 46232485 EC50 = 316.23 nM T86273 CU3YK2 46232486 EC50 = 316.23 nM T86273 CV20ZY 46232487 EC50 = 3981.07 nM T86273 C87MOU 46232488 EC50 = 12589.25 nM T86273 CHZX09 46232489 EC50 > 7943.28 nM T86273 CY9ED0 46232528 EC50 = 7943.28 nM T86273 CD78SA 46232529 EC50 = 158.49 nM T86273 CQBX08 46232530 EC50 = 7.943 nM T86273 CN62KF 46232531 EC50 = 501.19 nM T86273 CYE8W7 46232532 EC50 = 12.59 nM T86273 CJ7WT0 46232566 EC50 = 12.59 nM T86273 CCB75O 46232567 EC50 = 12.59 nM T86273 C4IW3T 46232568 EC50 = 79.43 nM T86273 CJ6FH7 46232569 EC50 = 1000 nM T86273 C0PGE7 46232570 EC50 = 63.1 nM T86273 CUH8W5 46232571 EC50 = 1 nM T86273 CK5UF1 46232594 EC50 = 5011.87 nM T86273 CZ3JW0 46232595 EC50 = 31.62 nM T86273 C2ES4M 46232596 EC50 = 316.23 nM T86273 CQVX29 46232597 EC50 = 1258.93 nM T86273 CRBJ17 46232598 EC50 = 19.95 nM T86273 CA16WL 46232626 EC50 = 630.96 nM T86273 C81AMZ 46232627 EC50 = 630.96 nM T86273 CAER49 46232628 EC50 = 31.62 nM T86273 C35TJS 46232629 EC50 = 39.81 nM T86273 C47NSZ 46232656 EC50 = 316.23 nM T86273 CC7TB2 46232657 EC50 = 3162.28 nM T86273 CQ8Y9L 46232658 EC50 = 1258.93 nM T86273 C3PKO0 46232659 EC50 = 3.981 nM T86273 C8NYM1 46232660 EC50 = 19.95 nM T86273 CD5A1X 46232694 EC50 = 10 nM T86273 CW46RF 46232695 EC50 = 3.981 nM T86273 CE9V5S 46232696 EC50 = 10 nM T86273 C3ISH8 46232697 EC50 = 794.33 nM T86273 CM7VX3 46232698 EC50 = 3162.28 nM T86273 CC05HT 46232736 EC50 = 12.59 nM T86273 CL25UR 46232737 EC50 = 63.1 nM T86273 CL5EJ4 46232875 EC50 = 1258.93 nM T86273 C1YBO4 46232982 EC50 = 398.11 nM T86273 C7UKJ1 46232983 EC50 = 2511.89 nM T86273 CNYC06 46232984 EC50 = 630.96 nM T86273 CAR63C 46232985 EC50 = 501.19 nM T86273 C1A9DH 46232986 EC50 = 1995.26 nM T86273 CU8J9L 46233020 EC50 = 630.96 nM T86273 C0YED6 46233021 EC50 = 15.85 nM T86273 CGY7E3 46233022 EC50 = 125.89 nM T86273 CY2X6C 46233023 EC50 = 398.11 nM T86273 CK1V4A 46233024 EC50 = 1258.93 nM T86273 CP2TZ5 46233052 EC50 = 125.89 nM T86273 CW0EC5 46233053 EC50 = 2511.89 nM T86273 CDXC43 46233054 EC50 = 63.1 nM T86273 CDF5L9 46233055 EC50 = 251.19 nM T86273 C2SND5 46233056 EC50 = 100 nM T86273 CSDU94 52905075 EC50 = 17200 nM T86273 C8R2XS 52941296 IC50 = 6900 nM T86273 CG0EB8 52941356 IC50 = 880 nM T86273 C8UCO4 52941357 IC50 = 1100 nM T86273 CPS8U6 52941381 IC50 = 5500 nM T86273 CA1YS7 52942648 IC50 > 10000 nM T86273 CH8R3Y 52943980 IC50 > 10000 nM T86273 CQG3X0 52945144 IC50 = 500 nM T86273 CR1JQ2 52945302 IC50 = 11000 nM T86273 CV7D9R 52945575 IC50 > 10000 nM T86273 CM7OH6 52946134 IC50 = 4500 nM T86273 CN8V0Y 52946277 IC50 = 82 nM T86273 CLIE05 52946355 IC50 = 710 nM T86273 C1J7ZR 52946791 IC50 = 430 nM T86273 C5Y1NH 52947341 IC50 = 5000 nM T86273 C3UA5E 52947397 IC50 > 10000 nM T86273 CBD79A 52948571 IC50 = 2700 nM T86273 C0MTQ6 52948780 IC50 = 580 nM T86273 C05MNR 52948858 IC50 = 5000 nM T86273 CL52ZT 52949831 IC50 > 10000 nM T86273 CU24VT 52949938 IC50 = 2800 nM T86273 C9VM8U 52950002 IC50 = 490 nM T86273 C89QMJ 53311618 EC50 = 48 nM T86273 CQ9HO5 53311701 EC50 = 3.5 nM T86273 C9GZ1T 53311781 EC50 = 49 nM T86273 CC16MD 53311869 EC50 = 1.5 nM T86273 C49KBY 54586161 EC50 = 55000 nM T86273 C7NA3K 59053728 EC50 > 10000 nM T86273 C5VS9J 66668687 EC50 > 10000 nM T86273 CQ95HE 66737876 EC50 = 220 nM T86273 C15VPJ 66739980 EC50 = 17.08 nM T86273 CY3QR9 66740913 EC50 = 470 nM T86273 CD4IA7 67922813 EC50 = 1050 nM T86273 CK6FY9 70682209 EC50 = 160000 nM T86273 C7OQ1W 70682210 EC50 = 650 nM T86273 CG3N5L 70684311 EC50 = 25000 nM T86273 CFSI97 70686469 EC50 = 87000 nM T86273 C0ZK8Y 71450251 EC50 = 0.72 nM T86273 C2YPG5 71450252 EC50 = 2.8 nM T86273 C3KYD0 71452075 EC50 = 47 nM T86273 CMNU91 71452076 EC50 = 23 nM T86273 C2ZOV4 71452077 EC50 = 127 nM T86273 C81PWI 71452078 EC50 = 20 nM T86273 C02OJU 71452079 EC50 = 30 nM T86273 CLS12C 71452080 EC50 = 2.9 nM T86273 C1XPG6 71453901 EC50 = 6.2 nM T86273 C78WKX 71453902 EC50 = 3151 nM T86273 C1K3DR 71453903 EC50 > 10000 nM T86273 CV7N8X 71453904 EC50 = 5422 nM T86273 CGW25V 71453905 EC50 = 3871 nM T86273 C6NT5L 71453906 EC50 = 710 nM T86273 C5E0GQ 71455632 EC50 = 12 nM T86273 C3WL6V 71455633 EC50 = 12 nM T86273 C09TYE 71455634 EC50 = 0.46 nM T86273 C7X4PJ 71455635 EC50 = 3711 nM T86273 CK3ZA5 71455636 EC50 = 30 nM T86273 CJUB17 71457417 EC50 = 4886 nM T86273 CJ1UZ8 71457418 EC50 = 12 nM T86273 CRIX26 71457419 EC50 > 10000 nM T86273 CMK0J6 71459273 EC50 = 27 nM T86273 C43HJS 71459274 EC50 = 7.9 nM T86273 C9DL0W 71459275 EC50 = 3.1 nM T86273 CMIF69 71459276 EC50 = 7.1 nM T86273 CM3RX0 71461053 EC50 = 451 nM T86273 C79HLK 71461054 EC50 = 0.72 nM T86273 C3NBR7 71461055 EC50 = 69 nM T86273 CP3KO8 71461056 EC50 = 535 nM T86273 C56PNW 71461057 EC50 = 160 nM T86273 CRQV93 71461058 EC50 = 590 nM T86273 C0TF5J 71462786 EC50 = 0.6 nM T86273 C9BU3G 71462787 EC50 = 0.31 nM T86273 CB54JL 71462788 EC50 = 164 nM T86273 C67ZSQ 71540073 EC50 = 2.3 nM T86273 CJ0UR1 71540074 EC50 = 1.6 nM T86273 C7DZA6 71540075 EC50 = 4.7 nM T86273 CV8G2U 71540076 EC50 = 2.7 nM T86273 C4YX0D 71540077 EC50 = 43 nM T86273 CSE3H2 71540078 EC50 = 2 nM T86273 CPK6M4 71540174 EC50 = 3.3 nM T86273 C1SWJ2 71540175 EC50 = 2.8 nM T86273 CHDC40 71541719 EC50 = 2.5 nM T86273 C1IP4Y 71541720 EC50 = 257 nM T86273 C3O6FA 71541721 EC50 = 78 nM T86273 CFZ41A 71541722 EC50 = 9.2 nM T86273 C4EQ8L 71541723 EC50 = 137 nM T86273 CC3YK0 71559936 EC50 = 337 nM T86273 CU4QO1 71559937 EC50 = 349 nM T86273 CO9U3K 71561365 EC50 = 15 nM T86273 CXY59Q 71561366 EC50 = 7.9 nM T86273 CV96QS 71561367 EC50 = 65 nM T86273 CDCG91 71561368 EC50 = 12 nM T86273 CXZ6G1 71561369 EC50 = 1480 nM T86273 CVBM25 71561370 EC50 = 113 nM T86273 C43ZMU 71561499 EC50 = 2910 nM T86273 CGV02W 71561500 EC50 = 4930 nM T86273 C2SI5W 71561501 EC50 > 10000 nM T86273 C0XGB5 71561502 EC50 = 920 nM T86273 CAK36Y 71561503 EC50 > 10000 nM T86273 CS6M9T 71561504 EC50 = 6.8 nM T86273 C2KC8U 71561614 EC50 = 15 nM T86273 CW5G6L 71561615 EC50 = 4680 nM T86273 CZ0NA6 71561616 EC50 = 9530 nM T86273 C1EI7U 71561617 EC50 = 3140 nM T86273 CP3M6F 71561618 EC50 = 1400 nM T86273 CT52NW 71561619 EC50 = 393 nM T86273 C6BRT4 71561751 EC50 > 10000 nM T86273 CR6O2T 71561752 EC50 > 10000 nM T86273 CCR2N8 71561753 EC50 = 1.2 nM T86273 C8M6WR 71561754 EC50 = 0.3 nM T86273 CMR24O 71561755 EC50 = 1.8 nM T86273 CM2DR4 71561756 EC50 = 1.2 nM T86273 CO8HJ4 71561881 EC50 = 6400 nM T86273 CZ1SK4 71561882 EC50 = 2.4 nM T86273 CPF32W 71561883 EC50 = 14 nM T86273 CV84NI 71561884 EC50 = 7.9 nM T86273 CW34IF 71561885 EC50 = 18 nM T86273 C2N5WV 71599441 EC50 = 125.89 nM T86273 CBQ7V8 71626228 EC50 = 5000 nM T86273 C7SC5R 71626229 EC50 = 15000 nM T86273 CP8RB5 71626232 EC50 = 378000 nM T86273 CIQ6O5 71626422 EC50 = 240 nM T86273 C0CU1B 71626488 EC50 = 1.5 nM T86273 C02GPL 71626489 EC50 = 17 nM T86273 CWRE16 71626490 EC50 = 41 nM T86273 C4T0YO 71626491 EC50 = 162 nM T86273 CA5Q7Y 71626492 EC50 = 10.7 nM T86273 CS91PQ 71626493 EC50 = 59 nM T86273 CRY4K3 71626555 EC50 = 64 nM T86273 CIC2R3 71626556 EC50 = 25 nM T86273 C5RCJ7 71626557 EC50 = 40 nM T86273 C0GZM5 71626558 EC50 = 148 nM T86273 C2YAL3 71626559 EC50 = 1216 nM T86273 CZ0X6R 71626560 EC50 = 15 nM T86273 CKF0W7 71626697 EC50 = 16 nM T86273 C6A4KG 71626699 EC50 = 0.45 nM T86273 C25GST 71626700 EC50 = 1.4 nM T86273 CC1J3T 71626765 EC50 = 3800 nM T86273 CJK28X 71626832 EC50 = 35000 nM T86273 CH76KG 71626833 EC50 = 12000 nM T86273 CQ6K7S 71626834 EC50 = 8000 nM T86273 CZ8DO6 71626905 EC50 = 5300 nM T86273 C58NVG 71660821 EC50 = 25.12 nM T86273 C2QC6B 71660822 EC50 = 316.23 nM T86273 CQ92NT 71660823 EC50 = 251.19 nM T86273 CEK50W 71660856 EC50 = 3981.07 nM T86273 CK2NI9 71660881 EC50 > 10000 nM T86273 C2BE9R 71660884 EC50 > 10000 nM T86273 CX2KL4 71660910 EC50 = 1000 nM T86273 C3QT0P 71660960 EC50 = 125.89 nM T86273 C12HBK 71660979 EC50 = 63.1 nM T86273 CDZ5F6 71661092 EC50 = 100 nM T86273 C7FX6P 71661185 EC50 = 50.12 nM T86273 CYM6K1 71661186 EC50 = 199.53 nM T86273 C3FB6C 71661220 EC50 = 199.53 nM T86273 CCV37X 71661222 EC50 = 1584.89 nM T86273 CJNK51 71661223 EC50 = 2511.89 nM T86273 CC24DT 71661224 EC50 = 1000 nM T86273 CR03WD 71691935 EC50 = 5080 nM T86273 CT6IL4 71718878 EC50 = 5.5 nM T86273 C68XHQ 71720725 EC50 = 120 nM T86273 CK15QE 71812800 EC50 > 10000 nM T86273 C6NQ0W 73346390 EC50 = 892 nM T86273 C3BXT6 73346391 EC50 = 7430 nM T86273 C2PL1B 73347897 EC50 = 61 nM T86273 C2A4CJ 73347898 EC50 = 1270 nM T86273 C04TUI 73349425 EC50 = 384 nM T86273 C34QED 73349426 EC50 = 63 nM T86273 CBVL49 73349428 EC50 = 500 nM T86273 CSU3M8 73350992 EC50 = 204 nM T86273 C96LOS 73350993 EC50 = 466 nM T86273 C30IAY 73350994 EC50 = 260 nM T86273 CQ5P4C 73350995 EC50 = 120 nM T86273 C0I1QR 73352462 EC50 = 440 nM T86273 C3XU8Z 73352464 EC50 = 580 nM T86273 CFO79G 73352466 EC50 = 35 nM T86273 CY86ES 73352467 EC50 = 62 nM T86273 C6V2NJ 73353937 EC50 = 53 nM T86273 C5V4BH 73353938 EC50 = 406 nM T86273 CB41UL 73353940 EC50 = 31 nM T86273 CDH70E 73353941 EC50 = 32 nM T86273 C7BHF0 73353942 EC50 = 4080 nM T86273 CRN0Z4 73353943 EC50 = 310 nM T86273 CV3J8S 73353944 EC50 = 1230 nM T86273 C4BYW2 73355479 EC50 = 910 nM T86273 C56RNJ 73355480 EC50 = 350 nM T86273 COF7Q1 73355481 EC50 = 470 nM T86273 C2M3OK 73357023 EC50 = 458 nM T86273 CG2ID5 73357024 EC50 = 51 nM T86273 CX3R5Z 73357025 EC50 = 2100 nM T86273 CA92FL 73357026 EC50 = 320 nM T86273 CSFR42 74766512 EC50 = 390 nM T86273 C6QB2C 76314787 EC50 = 1.9 nM T86273 CL3AZ9 76314788 EC50 = 102 nM T86273 C6WT0P 76314983 EC50 > 100000 nM T86273 C0QX8M 76318386 EC50 = 10 nM T86273 CGO85D 76318387 EC50 = 8.2 nM T86273 C9QDT4 76322064 EC50 = 2.1 nM T86273 CPV2F6 76322065 EC50 = 160 nM T86273 C87MUN 76328184 EC50 = 1320 nM T86273 CEQZ97 76332905 EC50 = 135 nM T86273 COS64J 76336516 EC50 = 11 nM T86273 CP2D1Y 77845059 EC50 = 1.7 nM T86273 CG8VY9 77845211 EC50 = 1358 nM T86273 C5FT1B 77845284 EC50 = 675 nM T86273 CARX24 77846087 EC50 = 7.7 nM T86273 CF1U0T 89501377 EC50 > 1000 nM T86273 CSC4O3 89501409 EC50 = 1.6 nM T86273 CL2V1Q 89501422 EC50 = 21.6 nM T86273 C8P3OG 89501425 EC50 = 67.5 nM T86273 CKP79C 89501429 EC50 = 2.3 nM T86273 C8O0IW 89501434 EC50 = 14.4 nM T86273 C1JOZ9 89501446 EC50 = 0.057 nM T86273 CA3CS5 89501494 EC50 = 7.8 nM T86273 C4SYV7 89501496 EC50 > 100 nM T86273 C4U3KM 89501521 EC50 = 19.6 nM T86273 C5Y7MH 89501534 EC50 > 100 nM T86273 CWF26V 89501566 EC50 > 100 nM T86273 CY4U5T 89501594 EC50 = 5.8 nM T86273 CQRS86 89501598 EC50 > 1000 nM T86273 C94TUF 89501608 EC50 = 16.8 nM T86273 CPG39S 89501618 EC50 = 94.7 nM T86273 C5TA3Q 89501664 EC50 = 35.7 nM T86273 CG90MO 89501666 EC50 = 1.48 nM T86273 CRC6J5 89501780 EC50 = 38 nM T86273 CSN2U6 89501844 EC50 = 8.6 nM T86273 CDY15Z 89501851 EC50 = 17.2 nM T86273 C1W0SN 89651284 EC50 = 794.33 nM T86273 CX0H4A 89707030 EC50 = 3050 nM T86273 CUO1D7 90283905 EC50 = 9130 nM T86273 CGZT28 90284086 EC50 = 580 nM T86273 CIL04D 90284520 EC50 = 730 nM T86273 CGQW57 90327488 EC50 = 63 nM T86273 CMA90I 90327533 EC50 = 119 nM T86273 CYU01J 90644444 EC50 = 18 nM T86273 CT5SW3 90644445 EC50 = 78 nM T86273 C7FW1D 90644446 EC50 = 24 nM T86273 CF9OW0 90644447 EC50 = 30 nM T86273 C5GQ0W 90644448 EC50 = 35 nM T86273 CWQ97Z 90644449 EC50 = 178 nM T86273 CECW26 90644450 EC50 = 520 nM T86273 CX69CY 90644451 EC50 = 0.28 nM T86273 C57SRN 90644452 EC50 = 2.3 nM T86273 CJY69M 90644453 EC50 = 5.2 nM T86273 CF6C5U 90644454 EC50 = 5.5 nM T86273 CPW29U 90644455 EC50 = 8.5 nM T86273 C64BWS 90644456 EC50 = 8.9 nM T86273 C9OWV0 90644457 EC50 = 34 nM T86273 CHK47R 90644458 EC50 = 25 nM T86273 CTA54R 90644459 EC50 = 38 nM T86273 C2LAH8 90644460 EC50 = 1405 nM T86273 C6AU0Q 90654563 EC50 = 20 nM T86273 CSW57N 90654564 EC50 = 8 nM T86273 CY8VB0 90654565 EC50 = 274 nM T86273 CK8J1R 90654566 EC50 = 4 nM T86273 C7R8YB 90654567 EC50 > 8000 nM T86273 C23TZB 90654568 EC50 = 19 nM T86273 C1PXV9 90654569 EC50 = 60 nM T86273 CXP47I 90654570 EC50 = 320 nM T86273 C2R1QN 90654571 EC50 = 33 nM T86273 CLQ1I7 90654572 EC50 = 4300 nM T86273 C3S0HW 90654573 EC50 = 95 nM T86273 C15NGP 90654574 EC50 = 8 nM T86273 C49RES 90654575 EC50 = 930 nM T86273 C1YN6P 90654576 EC50 = 13700 nM T86273 CG5MP2 90654577 EC50 = 2100 nM T86273 C4VSK5 90654578 EC50 = 220 nM T86273 CQJC26 90654579 EC50 = 930 nM T86273 C3SLF4 90654580 EC50 = 13 nM T86273 CHQ6O4 90654581 EC50 = 17 nM T86273 COB1G5 90654582 EC50 = 140 nM T86273 C0KAP2 90654583 EC50 = 76 nM T86273 CY8CN2 90654584 EC50 = 2 nM T86273 CN8Y1A 90654585 EC50 = 4 nM T86273 C0XQB9 90654586 EC50 = 440 nM T86273 CHP74S 90654587 EC50 = 3 nM T86273 C12FTL 90654588 EC50 = 14 nM T86273 CYXW14 90654589 EC50 = 1 nM T86273 CPG7U1 90654590 EC50 = 6 nM T86273 CMB8C2 90654591 EC50 = 63 nM T86273 CLME72 90654592 EC50 = 38 nM T86273 CE4FM0 90654593 EC50 = 26 nM T86273 C3PH6W 90654594 EC50 = 12 nM T86273 CD4R6B 90654595 EC50 = 14 nM T86273 C3LBP4 90654596 EC50 = 30 nM T86273 CY3K5B 90654597 EC50 = 18 nM T86273 CT8PS3 90654598 EC50 = 11 nM T86273 C2ORH4 90654599 EC50 = 25 nM T86273 C96YCU 90654600 EC50 = 15 nM T86273 CQ78PX 90655903 EC50 = 200 nM T86273 C60SIF 91668293 EC50 = 4000 nM T86273 CM95VC 91758806 EC50 = 3.9 nM T86273 CBH2Y4 91972025 EC50 = 440 nM T86273 C7R6IK 101882290 EC50 = 30000 nM T86273 C4HM9W 101882379 EC50 = 17200 nM T86273 CNJ2G6 101886302 EC50 = 1030 nM T86273 CC3PM5 101886309 EC50 = 400 nM T86273 CW27MY 118063735 EC50 > 80000 nM T86273 CU7CX8 118093390 EC50 = 199.53 nM T86273 CR57JD 118093402 EC50 = 158.49 nM T86273 CNH12F 118093410 EC50 = 125.89 nM T86273 CF9O1R 118093418 EC50 = 1995.26 nM T86273 C1T2AY 118093420 EC50 = 199.53 nM T86273 C7Z8QO 118093441 EC50 = 1000 nM T86273 C1PO5A 118093476 EC50 = 79.43 nM T86273 CVZP24 118093484 EC50 = 316.23 nM T86273 C8NBJ2 118093493 EC50 = 125.89 nM T86273 CQ1NY5 118093506 EC50 = 794.33 nM T86273 CWA34K 118093510 EC50 = 251.19 nM T86273 C0MOW7 118093511 EC50 = 7943.28 nM T86273 CEK45C 118093535 EC50 = 31.62 nM T86273 C5U6ZY 118093541 EC50 = 63.1 nM T86273 C89CQL 118093557 EC50 = 25.12 nM T86273 CN2MY9 118093562 EC50 = 50.12 nM T86273 C6I5PO 118093575 EC50 = 100 nM T86273 CJ49IZ 118093582 EC50 = 39.81 nM T86273 C9DUO5 118103668 EC50 = 100 nM T86273 C80VXA 118103672 EC50 = 31.62 nM T86273 C6IPM5 118103673 EC50 = 398.11 nM T86273 CD6EG0 118103679 EC50 = 100 nM T86273 C6QIR5 118103697 EC50 = 79.43 nM T86273 CUZ8R7 118103698 EC50 = 25.12 nM T86273 CCV78A 118103700 EC50 = 100 nM T86273 CBC9J6 118103718 EC50 = 398.11 nM T86273 CVNA28 118103734 EC50 = 100 nM T86273 C0MWT9 118103736 EC50 = 501.19 nM T86273 CFE4I9 118103740 EC50 = 199.53 nM T86273 C1L2QX 118104381 EC50 = 251.19 nM T86273 CC9E1T 118104385 EC50 = 794.33 nM T86273 CIXV65 118104397 EC50 = 251.19 nM T86273 CH30QC 118455116 EC50 > 50000 nM T86273 C8JKB0 118455158 EC50 = 12500 nM T86273 CZ1UG7 118455177 EC50 > 50000 nM T86273 CDV93J 118455249 EC50 > 50000 nM T86273 C8XSY9 118455251 EC50 > 50000 nM T86273 CKW02O 118464620 EC50 > 50000 nM T86273 C1M6HI 118464622 EC50 = 35180 nM T86273 CZ90CS 118464628 EC50 > 50000 nM T86273 CQ8FZ1 118464629 EC50 > 50000 nM T86273 C9Z5IS 118464630 EC50 > 50000 nM T86273 CE8IB7 118464638 EC50 = 1880 nM T86273 CBMC28 118464639 EC50 > 50000 nM T86273 C0O9KA 118464662 EC50 = 25100 nM T86273 CC94VK 118464664 EC50 = 680 nM T86273 CS4FG3 118464680 EC50 = 3400 nM T86273 C2LW6I 118464701 EC50 > 50000 nM T86273 CFT41Z 118464713 EC50 > 50000 nM T86273 C98JGK 118464718 EC50 = 3500 nM T86273 C1A7LK 118464720 EC50 > 50000 nM T86273 C5N4KZ 118464724 EC50 = 20500 nM T86273 C7T0LW 118464729 EC50 > 50000 nM T86273 CKDR72 118464738 EC50 > 50000 nM T86273 C0M1HP 118464746 EC50 > 50000 nM T86273 CTFI52 118464747 EC50 = 930 nM T86273 C14BUX 118464749 EC50 > 50000 nM T86273 CSK23C 118464755 EC50 > 50000 nM T86273 C85QJC 118464758 EC50 = 30500 nM T86273 C2GFK9 118464786 EC50 > 50000 nM T86273 CZ29VE 118464802 EC50 > 50000 nM T86273 CKZ46Y 118464803 EC50 = 770 nM T86273 COR17F 118464804 EC50 = 1400 nM T86273 C5R0GL 118464805 EC50 > 50000 nM T86273 CZU2T0 118464806 EC50 = 15800 nM T86273 CL2C3U 118464811 EC50 = 3730 nM T86273 CUR6C2 118464815 EC50 = 4308 nM T86273 C4MHL0 118464823 EC50 > 50000 nM T86273 CVY96U 118576916 EC50 = 299 nM T86273 CY3OZ8 118576930 EC50 = 20 nM T86273 CIR6K0 118576935 EC50 = 35 nM T86273 CI9XE6 118576958 EC50 = 35 nM T86273 C95IOA 118576974 EC50 = 128 nM T86273 C5AU2K 118576999 EC50 = 71 nM T86273 CO25TK 118577011 EC50 = 885 nM T86273 CXYB89 118577093 EC50 = 7745 nM T86273 CC27OP 118577297 EC50 = 260 nM T86273 C7RJS8 118577308 EC50 = 177 nM T86273 CN93ZX 118586274 EC50 > 10000 nM T86273 C8IS7P 118586276 EC50 = 994 nM T86273 CS40HD 118586278 EC50 = 254 nM T86273 C2XWO5 118586279 EC50 = 900 nM T86273 CLS69I 118586280 EC50 = 750 nM T86273 C2FZ1K 118586281 EC50 = 1106 nM T86273 CWGX59 118586282 EC50 = 4300 nM T86273 CQDW15 118586284 EC50 = 47 nM T86273 C2SHU6 118586298 EC50 = 156 nM T86273 C3SA1D 118709770 EC50 > 1000 nM T86273 C5YDM2 118709771 EC50 = 20 nM T86273 C4Z7EF 118709772 EC50 = 12 nM T86273 C74HYM 118709773 EC50 = 41 nM T86273 C2ZHY6 118709774 EC50 > 1000 nM T86273 CN01EP 118709775 EC50 > 1000 nM T86273 C3JEL7 118709776 EC50 = 178 nM T86273 CT1J7Y 118709777 EC50 = 5.1 nM T86273 CP9QJ6 118721858 EC50 = 122 nM T86273 C3D9EX 118725000 EC50 = 4390 nM T86273 COKI87 118728411 EC50 = 750 nM T86273 C7DS9W 118735265 EC50 = 9600 nM T86273 C4BI3X 118735266 EC50 = 30000 nM T86273 CLXS59 118735267 EC50 = 20000 nM T86273 CJB06R 118735268 EC50 = 25000 nM T86273 CE9H7Y 121322331 EC50 = 700 nM T86273 C2VU7H 121322333 EC50 = 315 nM T86273 CB6A8H 121355127 EC50 = 1770 nM T86273 CRAS43 122201312 EC50 = 205 nM T86273 CFBL98 126673445 EC50 = 337 nM T86273 CF1I5C 126673464 EC50 > 4500 nM T86273 C4KOS1 126673489 EC50 = 1113 nM T86273 CEW5F0 126673504 EC50 = 86 nM T86273 COE83Z 126700765 EC50 = 326 nM T86273 CJP3G0 127029731 EC50 = 31.5 nM T86273 CGYI50 130361811 EC50 = 1600 nM T86273 CCM3Z9 130361815 EC50 = 566 nM T86273 C87YAW 130361906 EC50 = 97.3 nM T86273 C4S8UI 130361919 EC50 = 1900 nM T86273 C1UJK4 130361936 EC50 = 3070 nM T86273 C34VCS 130361940 EC50 = 5380 nM T86273 C8DAE0 130361963 EC50 = 1380 nM T86273 CQ3JT2 130361991 EC50 = 8440 nM T86273 CZ6SC8 136002656 IC50 = 5100 nM T86273 CW23LV 136002657 IC50 > 10000 nM T86273 C1C2GL 136002658 IC50 > 10000 nM T86273 C6LR7Y 136167037 EC50 = 20 nM T86273 CE1KC2 137633639 EC50 >= 10000 nM T86273 CRM2F6 137634612 EC50 = 5680 nM T86273 CWJR14 137634963 EC50 = 21750 nM T86273 C5DQE4 137636275 EC50 = 20750 nM T86273 CK41YG 137636348 EC50 = 310 nM T86273 C4XP3H 137636567 EC50 = 24 nM T86273 CQGA98 137636635 EC50 > 50000 nM T86273 CFZ6I3 137638975 EC50 > 50000 nM T86273 CWQD36 137641119 EC50 = 16630 nM T86273 CX7J3R 137641988 EC50 = 29550 nM T86273 C2KDE9 137644372 EC50 = 77 nM T86273 CV0A8X 137645502 EC50 = 750 nM T86273 CACD18 137646020 EC50 > 50000 nM T86273 C6HZ9K 137646061 EC50 = 17800 nM T86273 CWQ6F0 137646769 EC50 > 50000 nM T86273 C56NEX 137649364 EC50 > 50000 nM T86273 CE21TH 137650298 EC50 = 238 nM T86273 CCH5W3 137651232 EC50 = 42620 nM T86273 CPB80D 137651596 EC50 > 50000 nM T86273 CEJG32 137653533 EC50 = 36800 nM T86273 CV70JW 137656785 EC50 > 50000 nM T86273 CBU45S 137656815 EC50 > 50000 nM T86273 CMD92N 137657436 EC50 > 50000 nM T86273 CS71VA 137660218 EC50 = 4940 nM T86273 CEJI38 137660534 EC50 > 50000 nM T86273 CZS5G8 137661039 EC50 = 8260 nM T86273 C4DVO7 137661958 EC50 > 50000 nM T86273 C6A8TR 145177795 EC50 = 240 nM T86273 CPZX74 145949879 EC50 = 280 nM T86273 C5S9DQ 145955411 EC50 = 420 nM T86273 C1L3NH 145955827 EC50 = 160 nM T86273 CYS2J3 145956445 EC50 = 240 nM T86273 CXK82F 145961505 EC50 > 100 nM T86273 CX58KF 145962358 EC50 = 2.3 nM T86273 CN28EV 145967535 EC50 = 63.1 nM T86273 CA2FI0 145971348 EC50 = 39.81 nM T86273 CED8N1 145972818 EC50 = 100 nM T86273 CA6U8M 145973129 EC50 = 520 nM T86273 C0DEA1 145974037 EC50 = 31.62 nM T86273 CMD72S 145975890 EC50 = 79.43 nM T86273 C8FG5D 145978106 EC50 = 125.89 nM T86273 C5VT6H 155339362 EC50 = 10.5 nM T86273 CHQG81 155339372 EC50 = 5.59 nM T86273 CU6S9P 155528730 EC50 = 19900 nM T86273 CN05RX 155534242 EC50 = 223 nM T86273 CBW0S9 155534680 EC50 = 2770 nM T86273 C10HEY 155542354 EC50 > 30000 nM T86273 C8X7UQ 136166852 EC50 = 11 nM T86273 C0T4GZ 136166859 EC50 = 45 nM T86273 CK6VX4 136166933 EC50 = 12 nM T86273 CI3Q5M 136166936 EC50 = 23 nM T86273 CBGQ25 136166950 EC50 = 57 nM T86273 C3TM5W 136166952 EC50 = 100 nM T86273 CXOF15 136166966 EC50 = 25 nM T86273 C4WO9T 136167004 EC50 = 4 nM T86273 C0VP9J 136260512 EC50 = 380 nM T86273 D00QPU 12594 EC50 = 127000 nM T86273 D00WBS 3035026 EC50 = 1180 nM T86273 D02CWP 439763 EC50 = 290 nM T86273 D02YJL 387316 EC50 = 1920 nM T86273 D03RKW 9848818 EC50 = 30000 nM T86273 D05KJY 72326 EC50 > 10000 nM T86273 D06RBG 5283906 EC50 = 270 nM T86273 D07LUJ 64945 EC50 = 1430 nM T86273 D08WQV 10140 EC50 = 13600 nM T86273 D09MWG 5880 EC50 = 3760 nM T86273 D09OWE 92802 EC50 > 10000 nM T86273 D0AS9Q 12310288 EC50 = 33900 nM T86273 D0B7AH 45483949 EC50 = 166 nM T86273 D0D8IS 12544 EC50 = 3880 nM T86273 D0LC7K 119034 EC50 > 10000 nM T86273 D0SJ2Q 10494 EC50 = 2250 nM T17687 D01PZD 5329098 IC50 = 5000 nM T17687 D0B0AX 5328127 IC50 = 60 nM T17687 D0E3TC 44259 IC50 = 420 nM T17687 D0M9QZ 11485656 IC50 = 12500 nM T17687 D0Q7RE 16007391 Ki > 10000 nM T17687 D0VF6E 1401 IC50 = 7 nM T17687 D04FHB 6918852 Ki > 5000 nM T17687 D0H8KG 5311382 IC50 = 44 nM T17687 D0IT6Q 3038522 IC50 = 170 nM T17687 D0L5YF 5329032 IC50 = 1500 nM T17687 D0Z0KD 5330258 IC50 = 8620 nM T17687 CH21PG 2428 IC50 > 50000 nM T17687 CRFU83 156413 IC50 > 50000 nM T17687 C30UNK 247352 IC50 = 4700 nM T17687 C8HXQ5 247358 IC50 = 4200 nM T17687 CWGJ94 256524 Ki = 23000 nM T17687 CU5B1Z 4369491 IC50 > 50000 nM T17687 CMC76E 5327864 IC50 = 1320 nM T17687 C43JFT 5327866 IC50 > 50000 nM T17687 CS0Q4N 5327875 IC50 > 50000 nM T17687 CI96EG 5327876 IC50 = 1970 nM T17687 CT86OE 5327877 IC50 = 1260 nM T17687 C23EZX 5327878 IC50 = 348 nM T17687 C3P8CG 5327885 IC50 = 510 nM T17687 CLH9Y3 5327908 IC50 = 48 nM T17687 CA7U3O 5327914 IC50 = 51 nM T17687 C5JI1A 5327917 IC50 = 61 nM T17687 CPT61U 5328112 IC50 = 130 nM T17687 CXR9K1 5328115 IC50 = 82 nM T17687 CM0H5O 5328117 IC50 = 400 nM T17687 CDM98R 5328125 IC50 = 780 nM T17687 CDY2O3 5328134 IC50 = 33 nM T17687 CC1O0M 5328135 IC50 = 48 nM T17687 COT45A 5328149 IC50 = 51 nM T17687 CF3AM9 5328157 IC50 = 125 nM T17687 CT9SO8 5328158 IC50 = 40 nM T17687 CJA36I 5328171 IC50 = 139 nM T17687 CDV19S 5328354 IC50 > 50000 nM T17687 C1D0YT 5328357 IC50 > 50000 nM T17687 CC4O6Y 5328360 IC50 > 50000 nM T17687 CWX63A 5329004 IC50 = 1 nM T17687 CJ68OQ 5329013 IC50 = 800 nM T17687 CB6V5Y 5329028 IC50 = 1700 nM T17687 C4VLR8 5329033 IC50 = 100 nM T17687 CLT7J9 5329034 IC50 = 3000 nM T17687 CSY10K 5329111 IC50 = 3710 nM T17687 C19GHD 5329117 IC50 > 50000 nM T17687 C8IF1G 5329132 IC50 = 1650 nM T17687 CE68LC 5329133 IC50 > 16000 nM T17687 CBS40G 5330125 IC50 = 150 nM T17687 CNWK81 5330126 IC50 = 4800 nM T17687 CV7GX5 5330127 IC50 = 1 nM T17687 CWAR90 5330128 IC50 = 2 nM T17687 CDG3Z1 5330129 IC50 = 3 nM T17687 C09VSN 5330130 IC50 = 0.4 nM T17687 CNMJ73 5330131 IC50 = 12000 nM T17687 CV4U8Y 5330132 IC50 = 2.6 nM T17687 C6D7WJ 5330133 IC50 = 560 nM T17687 C2UX4V 5330134 IC50 = 340 nM T17687 CH38FW 5330135 IC50 = 3 nM T17687 CWQ47D 5330136 IC50 = 2 nM T17687 CLI47K 5330157 IC50 = 2.7 nM T17687 CNI15R 5330158 IC50 = 6 nM T17687 C4IA7N 5330159 IC50 = 4 nM T17687 CW8G9J 5330166 IC50 = 15 nM T17687 C7Z2YH 5330167 IC50 = 6 nM T17687 CEX9A7 5330168 IC50 = 33 nM T17687 C3I6KF 5330169 IC50 = 37 nM T17687 C5PL8M 5330199 IC50 = 3295 nM T17687 COJ5A2 5330209 IC50 = 44200 nM T17687 CK02IH 5330226 IC50 = 6600 nM T17687 CG0P9J 5330228 IC50 = 5290 nM T17687 C4VGL1 5330252 IC50 = 70 nM T17687 C14OKG 5330256 IC50 = 51 nM T17687 C74GLB 5330264 IC50 > 5000 nM T17687 CL5I2U 5330279 IC50 = 1860 nM T17687 CUPQ08 6539985 IC50 = 4200 nM T17687 CMEZ23 6540005 IC50 = 1500 nM T17687 CHF7G5 9890746 IC50 = 160000 nM T17687 C2TC1L 9910609 IC50 = 29 nM T17687 C3EUB4 9911005 IC50 > 200000 nM T17687 CYW49X 9927718 IC50 > 25000 nM T17687 CHB0D2 9982235 IC50 = 7.3 nM T17687 C7Q5CN 10015651 IC50 = 5100 nM T17687 C1JUF8 10073832 IC50 = 21 nM T17687 CD7J3O 10231458 IC50 > 30000 nM T17687 CH30RC 10253133 IC50 > 10000 nM T17687 C6ZF0X 10386217 IC50 > 30000 nM T17687 C07XHY 10388612 IC50 = 4 nM T17687 C2VPT6 10436729 IC50 = 4.6 nM T17687 C95LYF 10457505 IC50 > 200000 nM T17687 C7PLI5 10478569 IC50 = 6.5 nM T17687 COB2X8 10602350 IC50 = 140 nM T17687 CJO8Q1 10738332 IC50 = 130 nM T17687 CJ4P5T 10905857 IC50 > 200000 nM T17687 CJ05CL 11048367 IC50 > 30000 nM T17687 COMB49 11155938 IC50 = 9.2 nM T17687 C2W5RC 11235063 IC50 > 50000 nM T17687 CC8J3N 11328182 IC50 = 46 nM T17687 CA6F4L 11352215 IC50 = 6.6 nM T17687 CG57WD 11374515 IC50 = 4.7 nM T17687 CX25IH 11407794 IC50 = 37 nM T17687 CQD35C 11419379 IC50 = 7.6 nM T17687 C7AI2V 11432911 IC50 = 130 nM T17687 C45WKC 11442803 IC50 = 1 nM T17687 CZ9O1A 11455031 IC50 = 44 nM T17687 CJUF06 11464544 IC50 = 54 nM T17687 CTG3D9 11465545 IC50 = 5.3 nM T17687 CE39WZ 11488852 IC50 = 33 nM T17687 CH2IZ9 11517688 IC50 = 10000 nM T17687 CU13WV 11518389 IC50 > 50000 nM T17687 CTG83F 11539329 Ki > 4700 nM T17687 CMIL86 11590363 Ki > 4700 nM T17687 C5B3XJ 11620410 IC50 = 4370 nM T17687 C9T6SC 11640926 Ki > 4700 nM T17687 C9P0VD 11729539 IC50 > 200000 nM T17687 CBCS71 12424767 IC50 = 25000 nM T17687 C3VY1T 15707182 IC50 = 9200 nM T17687 CFPW41 16007116 Ki > 4700 nM T17687 CL9BQ6 17748275 IC50 = 5360 nM T17687 CIYU37 44294299 IC50 = 126 nM T17687 CUE5J6 44294644 IC50 = 51 nM T17687 CW02AS 44294903 IC50 > 50000 nM T17687 CI93QN 44330124 IC50 = 10600 nM T17687 CCL6N3 44330125 IC50 = 15000 nM T17687 CK0DR6 44330126 IC50 = 6200 nM T17687 CMY49P 44330151 IC50 = 21000 nM T17687 C13ZHT 44330158 IC50 = 6800 nM T17687 C1U3NK 44330159 IC50 = 44000 nM T17687 CJ5KF3 44330203 IC50 = 5400 nM T17687 C5WP3Z 44390984 IC50 = 30 nM T17687 C54JRW 44399701 IC50 = 80 nM T17687 C7KZV2 44414322 IC50 = 34355 nM T17687 CJM06T 44414347 IC50 > 50000 nM T17687 CLS29B 46872626 IC50 > 10000 nM T17687 CM0U3I 155534552 IC50 = 573 nM T17687 D00HVA 11624601 Ki > 4700 nM T17687 D06LJL 9916282 IC50 = 8000 nM T17687 D09XIL 11396738 IC50 = 92 nM T17687 D0BW4G 10907042 IC50 = 29700 nM T17687 D0IR6U 5494425 IC50 = 1480 nM T17687 D0Q3NG 11715520 Ki > 4700 nM T17687 D0S7IE 11658882 Ki > 4700 nM T47306 CAHM60 9810725 IC50 = 1600 nM T47306 CK4JX7 9892294 IC50 = 210 nM T47306 CJ4W6B 10323324 IC50 = 2500 nM T47306 C39NFY 10370367 IC50 = 330 nM T47306 CY94NH 23661627 IC50 = 2500 nM T47306 CSD8Y2 23661628 IC50 = 2500 nM T47306 CL16CD 44434488 IC50 = 100000 nM T47306 CS6H9A 44434489 IC50 = 200000 nM T47306 CC92EV 44434491 IC50 = 12500 nM T47306 CZCM81 44434492 IC50 = 50000 nM T47306 CD2ZK1 44434504 IC50 = 50000 nM T47306 C1AG5X 44434506 IC50 = 20000 nM T47306 C26ZCX 44434507 IC50 = 5000 nM T47306 CBR3C8 44434508 IC50 = 20000 nM T47306 C80LUY 44434509 IC50 = 50000 nM T47306 CC39NE 54675753 IC50 = 200000 nM T47306 CGC2A6 90665602 IC50 = 80 nM T47306 CV3LY9 90665603 IC50 = 130 nM T47306 D02HCQ 1794427 IC50 = 226000 nM T47306 D0A9CK 9873573 IC50 = 3 nM T47306 D0HD2G 4788 IC50 = 340000 nM T47306 D0Z6OT 9850474 IC50 = 5 nM T24983 D01AZG 5073 Ki = 6.2 nM T24983 D01FFA 72301 Ki > 1000 nM T24983 D01ZII 2726 Ki = 25.12 nM T24983 D03QGM 5355 Ki = 2100 nM T24983 D05XGO 11154555 Ki = 110 nM T24983 D05ZIK 4205 Ki > 25 nM T24983 D06OSM 91273 Ki = 7.2 nM T24983 D07MEH 3033769 Ki = 3100 nM T24983 D08VRO 3822 Ki = 3.5 nM T24983 D09IOI 2170 Ki = 34 nM T24983 D0CQ0Z 33630 Ki = 1000 nM T24983 D0D1AL 3559 Ki = 0.74 nM T24983 D0G8NN 119570 Ki = 0.49 nM T24983 D0H3HM 60795 Ki = 57.1 nM T24983 D0H6QU 6005 EC50 = 4.3 nM T24983 D0H7KF 5002 Ki > 1000 nM T24983 D0I8FI 3779 Ki = 2900 nM T24983 D0J5RN 9690109 Ki > 100000 nM T24983 D0K8KX 5280343 Ki = 7846 nM T24983 D0KS6W 7077 Ki = 2765 nM T24983 D0R1JV 60854 Ki = 32 nM T24983 D0R6RO 4184 IC50 = 3311.31 nM T24983 D0R9EQ 5095 Ki = 7.8 nM T24983 D0T6QX 5736 Ki = 39 nM T24983 D0T7OW 681 Ki = 1.2 nM T24983 D0U5OE 3964 Ki = 4.9 nM T24983 D0V4QS 135398745 Ki = 19 nM T24983 D0WV3U 4893 Ki = 8300 nM T24983 D0X7KB 28864 EC50 = 88.5 nM T24983 D0X7QQ 16363 Ki = 0.066 nM T24983 D0Z1RV 135398737 Ki = 9 nM T24983 D01GEB 219050 Ki = 24 nM T24983 D0A7KI 3037308 Ki = 179 nM T24983 D0L3JI 188942 Ki = 3.6 nM T24983 D0LI1C 44469321 IC50 > 10000 nM T24983 D0N1HW 5311200 Ki = 0.4 nM T24983 D0W5EH 6918388 IC50 < 6 nM T24983 D0Y6HW 107930 Ki = 5515 nM T24983 D00MQS 9926143 IC50 = 1.3 nM T24983 D07YLK 4350931 Ki = 108 nM T24983 D00PXQ 60785 Ki = 2.9 nM T24983 D01PIL 54477 Ki = 3872 nM T24983 D01RAE 133079 Ki = 3.6 nM T24983 D02FNU 56971 IC50 = 1800 nM T24983 D02JMI 9888211 Ki = 79.43 nM T24983 D03TNA 5025739 EC50 = 12.4 nM T24983 D03ZZH 9887537 Ki = 10 nM T24983 D06DZI 107780 Ki < 10000 nM T24983 D07BCO 5684 Ki = 16 nM T24983 D0A3OF 10026300 IC50 = 150 nM T24983 D0EE6L 3038495 Ki = 38.9 nM T24983 D0K9JP 9928332 Ki = 234 nM T24983 D0M7LV 5761 Ki = 56 nM T24983 D0OS6O 60149 Ki = 11 nM T24983 D0OW1R 9802631 Ki = 2.1 nM T24983 D0T1SF 9909448 Ki > 3704 nM T24983 D0Z7AW 9820261 Ki = 3.4 nM T24983 C7ALK2 1240 Ki = 54 nM T24983 COJD92 1687 Ki = 1000 nM T24983 CXY0O5 4257 Ki = 0.03 nM T24983 C58GWB 4452 IC50 = 98.2 nM T24983 C5H9CN 9287 Ki > 10000 nM T24983 C3A6IG 16103 Ki = 420 nM T24983 C8OW9T 18519 Ki = 2500 nM T24983 C9E6DA 21171 Ki = 486 nM T24983 C87UJB 21454 Ki > 2600 nM T24983 CT60VY 32224 Ki = 0.54 nM T24983 C8Y6DE 37461 Ki = 185 nM T24983 CJS51G 52919 Ki = 5.8 nM T24983 CY2F8T 55445 Ki = 130 nM T24983 COI7E6 59227 Ki = 55 nM T24983 CBJ5R0 65340 Ki = 7.079 nM T24983 CK16NU 92716 Ki = 350 nM T24983 CN9GK1 104911 Ki = 16 nM T24983 C12BFY 114840 Ki = 3100 nM T24983 C9IBE6 125156 Ki > 3333 nM T24983 C5SWN1 127698 Ki = 90.9 nM T24983 CD2C0M 128054 Ki = 72 nM T24983 CN92EH 131396 Ki = 5 nM T24983 C1ND9W 161665 Ki > 1000 nM T24983 C9OD2N 163091 Ki = 9 nM T24983 CLK7P3 169713 IC50 > 10000 nM T24983 CRL1X5 178078 Ki = 61.4 nM T24983 CX39NY 188249 Ki = 109 nM T24983 C5RC4G 231915 Ki = 3 nM T24983 CM4E3I 233199 Ki = 250 nM T24983 CHZ1P6 380039 Ki = 352 nM T24983 CGZ34T 418856 Ki > 10000 nM T24983 CG2JX9 440229 Ki = 77.4 nM T24983 C28ARG 511482 Ki = 1.1 nM T24983 CG59VA 511484 Ki = 267 nM T24983 CS6X4W 667675 Ki = 20.4 nM T24983 CGIY90 688272 Ki = 2100 nM T24983 CU8H9L 749986 Ki = 94 nM T24983 CD7P8Y 763194 Ki = 57 nM T24983 C6QLR0 763343 Ki = 65 nM T24983 CLR75J 763625 Ki = 105 nM T24983 C5SXQ1 763774 Ki = 214 nM T24983 CW8R4B 778880 Ki = 2.2 nM T24983 C9IK2J 792265 Ki = 2 nM T24983 C13TYL 792460 Ki = 3.9 nM T24983 C4AY9X 792584 Ki = 0.7 nM T24983 CW0CU9 798232 Ki = 125.89 nM T24983 C9CZJ1 857428 Ki = 550 nM T24983 C2YWO6 863787 Ki = 88.9 nM T24983 CJ30IQ 1248739 Ki = 44 nM T24983 CM1TH8 1438298 Ki = 420 nM T24983 C0N4WD 1946142 Ki = 3 nM T24983 CJI01N 2099556 Ki = 9.6 nM T24983 C2H6TF 2653640 Ki = 0.7 nM T24983 C6N8EF 2812861 Ki = 8.5 nM T24983 CBWO62 2946349 Ki = 34 nM T24983 C64CZV 3038494 Ki = 44 nM T24983 CBL51N 3156990 Ki = 200 nM T24983 C82GMT 3246443 Ki = 1978 nM T24983 CXG36C 3428803 Ki = 59 nM T24983 C0U6EW 3504099 Ki = 0.03 nM T24983 CCH45N 3626837 Ki = 0.04 nM T24983 CD76NG 3691783 Ki = 3.6 nM T24983 CGZ02Q 3695490 Ki = 123 nM T24983 CK3W2U 3716121 Ki = 0.4 nM T24983 C9J5YC 3746693 Ki = 61 nM T24983 CI50PT 4064333 Ki = 162 nM T24983 CO0FZ1 4064342 Ki = 390 nM T24983 C1S6ZG 4088306 Ki = 18 nM T24983 CY7PH0 4302960 Ki = 63.1 nM T24983 CS6P5D 4797946 Ki = 1.89 nM T24983 CWV91F 4826074 Ki = 4.3 nM T24983 CWB9I2 4987774 Ki = 254 nM T24983 C6FM8G 5029739 Ki = 2.5 nM T24983 C9AZ2I 5249956 Ki = 134 nM T24983 CMX45W 5311346 Ki = 26.6 nM T24983 CYAT75 5493357 Ki = 145 nM T24983 C6L9DT 6466372 EC50 = 3.4 nM T24983 CWNZ35 6469693 Ki = 2.8 nM T24983 CJTQ40 6469918 EC50 = 1.8 nM T24983 CIZ7U3 6603820 EC50 = 17 nM T24983 CKP56W 6603867 Ki = 110 nM T24983 CSM9T8 6603950 Ki = 4.5 nM T24983 CW0ZE5 6918542 Ki > 3200 nM T24983 CC5PQ0 6918601 Ki > 3200 nM T24983 C1R4IO 6937303 Ki = 450 nM T24983 C6MR7E 8529065 Ki > 400 nM T24983 CZ1YG5 8592415 Ki = 39.1 nM T24983 C3NK0H 8690650 Ki = 91.8 nM T24983 CK3P4G 8704110 Ki = 61.9 nM T24983 C9R7NM 9104271 IC50 = 1.6 nM T24983 C8ZD1I 9129986 Ki = 9.9 nM T24983 CO40CQ 9794644 Ki = 228 nM T24983 CS05NC 9796180 Ki = 43 nM T24983 CUD06Z 9796627 Ki > 3900 nM T24983 CC5Z9T 9797161 IC50 = 17 nM T24983 CX3OB9 9797200 Ki = 24.5 nM T24983 CY6WB3 9797495 Ki = 1.1 nM T24983 CLUT03 9799123 Ki = 3 nM T24983 CEG5Z6 9799491 Ki > 1000 nM T24983 CZI29U 9799781 Ki = 4 nM T24983 CI4S6Y 9800164 Ki = 4 nM T24983 CFR7L3 9801098 Ki = 10 nM T24983 C5Z2KM 9805944 Ki = 1.1 nM T24983 C4MN6K 9815072 EC50 = 52 nM T24983 CV5L1J 9817253 Ki = 6.3 nM T24983 CJ78ZE 9817612 Ki = 1578 nM T24983 C6V0MU 9817774 Ki = 3.8 nM T24983 CWOS30 9817810 Ki > 3200 nM T24983 C12HJN 9818076 Ki = 31 nM T24983 C2V7HU 9819770 Ki = 8.8 nM T24983 C0XE2V 9820048 Ki = 100 nM T24983 CQE93H 9820085 Ki = 20.8 nM T24983 C3JBY9 9820304 Ki = 5 nM T24983 CR17LP 9820313 Ki = 37 nM T24983 C1HNW6 9820680 Ki = 7 nM T24983 C9D4HQ 9821010 Ki = 3.2 nM T24983 COJ3V6 9821803 Ki = 5 nM T24983 C0AU9L 9826801 Ki = 4300 nM T24983 C2F5OX 9828632 Ki = 65 nM T24983 CD64HG 9835713 EC50 = 12 nM T24983 CG40WZ 9836209 EC50 = 64 nM T24983 C6IX0Q 9836662 EC50 = 13.9 nM T24983 COG0R8 9836900 Ki = 6.1 nM T24983 CO7HQ5 9837137 Ki = 170 nM T24983 CX2OY0 9838927 EC50 = 228 nM T24983 C4BPW7 9839426 Ki = 4.9 nM T24983 C8XER9 9840365 Ki = 2 nM T24983 CI62VW 9840412 Ki = 14 nM T24983 C1U6ZX 9840672 Ki = 3.1 nM T24983 C8XFV5 9840797 Ki = 59 nM T24983 C6Z0GS 9841249 Ki = 14 nM T24983 CF87HQ 9841608 Ki = 27.8 nM T24983 CWPC68 9842859 Ki = 558 nM T24983 CR31XS 9843031 Ki = 47 nM T24983 CKZ0X3 9843032 Ki = 96 nM T24983 CN09KS 9843137 Ki = 429 nM T24983 C5MHS3 9847013 Ki = 2.3 nM T24983 C21SZB 9848933 Ki > 1000 nM T24983 CU52WK 9857248 EC50 = 10.1 nM T24983 CIV9L3 9857887 EC50 = 8 nM T24983 CN3Y0G 9858141 EC50 = 14.6 nM T24983 C7EZ2L 9859861 EC50 = 9 nM T24983 CT78EC 9860183 Ki = 2 nM T24983 C4GT3Z 9861459 Ki = 7 nM T24983 CD12MS 9861786 Ki = 15.8 nM T24983 CNCK78 9862256 Ki > 3200 nM T24983 C4YA9P 9863108 Ki = 12.59 nM T24983 C8M5XK 9863333 Ki = 2.4 nM T24983 C9A4PH 9865446 Ki = 11 nM T24983 C1SM8I 9865490 Ki = 5 nM T24983 C5WYN4 9865858 Ki = 70.9 nM T24983 CWN76A 9865920 Ki = 701 nM T24983 C7EX8O 9867004 Ki = 36 nM T24983 C4IZ3J 9867233 Ki = 5 nM T24983 CB1F0C 9867475 Ki > 3200 nM T24983 CDFP50 9868793 IC50 = 1102 nM T24983 CQ4LC2 9872676 Ki = 2510 nM T24983 C96CAU 9879627 EC50 = 36.2 nM T24983 CA7Y1H 9881000 EC50 = 86 nM T24983 CY5HZ0 9882594 Ki = 92 nM T24983 CJL1X0 9883552 Ki = 27 nM T24983 COI69G 9883554 Ki = 23.99 nM T24983 CW97YN 9883587 Ki = 1.5 nM T24983 C2GU0S 9884771 Ki = 75 nM T24983 CTAC24 9885114 Ki = 4.3 nM T24983 COT4C7 9885219 Ki = 106 nM T24983 C1FG7S 9886340 Ki = 48 nM T24983 CALV92 9886609 Ki = 73 nM T24983 CH84KI 9887091 Ki = 4.3 nM T24983 CYRS07 9887092 Ki = 7018 nM T24983 CJW1P5 9888494 Ki = 1230.27 nM T24983 C9GB2M 9888555 Ki = 15 nM T24983 C4PSF6 9888765 Ki = 0.55 nM T24983 C6WY0D 9891901 Ki = 3670 nM T24983 CAY10W 9901273 EC50 = 14.7 nM T24983 CBI9C5 9901894 IC50 = 5 nM T24983 CR8GO9 9902381 Ki = 4.3 nM T24983 C1U3EY 9902382 Ki = 10.7 nM T24983 C6RGI9 9904074 Ki = 272 nM T24983 CFI97S 9904205 IC50 = 131.83 nM T24983 CRLQ85 9905246 Ki = 21 nM T24983 CUN81Q 9905249 Ki = 1.3 nM T24983 C4QB8M 9905720 Ki = 32 nM T24983 CS2KM8 9906071 Ki = 16 nM T24983 CYWQ50 9906447 Ki > 10000 nM T24983 CD3F4N 9906454 Ki = 37.3 nM T24983 C7XS1O 9906895 Ki = 39 nM T24983 C7JFZ5 9906978 Ki = 3.6 nM T24983 C1SHO4 9907332 IC50 = 5.4 nM T24983 CDE29K 9907381 Ki = 3854 nM T24983 C07SWP 9907461 Ki = 10 nM T24983 CT96CK 9908071 Ki = 2469 nM T24983 C6YKE0 9908125 Ki = 22 nM T24983 CMZ58L 9909055 Ki = 14.2 nM T24983 CO7BK6 9909648 Ki = 3 nM T24983 C3BR6W 9910451 Ki = 920 nM T24983 C30JZT 9922161 EC50 = 44.8 nM T24983 CJL38X 9925730 Ki = 61.1 nM T24983 CG52QA 9926141 Ki = 311 nM T24983 CZ4WE9 9927411 Ki = 24 nM T24983 C4UYZ7 9927441 Ki > 3200 nM T24983 CMZF03 9928553 Ki = 93 nM T24983 CMS7Y8 9929581 Ki = 227 nM T24983 CB12RM 9929629 Ki = 2960 nM T24983 C2H8FQ 9930722 Ki = 1511 nM T24983 CN4HQ8 9930934 Ki = 21 nM T24983 CM3X7Y 9931571 Ki = 1760 nM T24983 C8BX2L 9945233 EC50 = 1 nM T24983 CAC12E 9945714 EC50 = 25 nM T24983 CS9O7H 9945753 EC50 = 3.9 nM T24983 C1ES5F 9946469 Ki = 6.9 nM T24983 CZPM75 9948461 Ki = 3.3 nM T24983 CO2DG9 9948546 Ki = 10 nM T24983 CU2JM9 9948584 Ki = 10 nM T24983 C9EUM1 9948965 Ki = 4.7 nM T24983 CO2QA0 9949442 Ki = 2.5 nM T24983 CA07XW 9949531 Ki = 11.2 nM T24983 COE2H3 9949554 Ki = 17 nM T24983 CIFG92 9949601 Ki = 12.4 nM T24983 C02IMR 9949655 IC50 = 3 nM T24983 CXEZ63 9950165 Ki = 0.6 nM T24983 CS95KP 9950913 Ki = 4377 nM T24983 C1K8WB 9951233 Ki = 4 nM T24983 CZ6D4W 9951735 Ki = 1 nM T24983 C8DQ6P 9952003 Ki = 5.4 nM T24983 C92UQN 9952218 Ki = 145 nM T24983 CHU17Z 9952528 Ki = 158.49 nM T24983 CWSE34 9954899 IC50 = 120 nM T24983 CL01HU 9966489 EC50 = 24 nM T24983 CZB52R 9967004 Ki = 18.3 nM T24983 CGP43F 9967140 IC50 = 8 nM T24983 CIW4R8 9968343 Ki = 5.1 nM T24983 CC1ZL3 9975465 Ki = 5.248 nM T24983 CXT1W6 9977478 Ki = 210 nM T24983 CMYN90 9977532 Ki = 0.23 nM T24983 CC6M7Z 9980998 Ki = 93 nM T24983 C4G1IX 9982854 Ki = 16.98 nM T24983 CP41ZO 9992499 Ki = 1647 nM T24983 CB2EP7 9995264 Ki = 3.6 nM T24983 CUS7W9 9995379 Ki = 3 nM T24983 CP31VK 9995904 Ki = 0.52 nM T24983 CWJ3C0 9997550 EC50 = 18 nM T24983 C7NC3D 10000302 Ki = 5.4 nM T24983 C6FA2J 10001207 Ki = 46 nM T24983 C8DM3P 10001519 Ki = 43 nM T24983 C0DIO1 10001810 Ki = 3 nM T24983 C1NQC9 10003809 Ki = 44.67 nM T24983 C27WPA 10007017 Ki = 602.56 nM T24983 CUX43N 10014136 Ki > 4067 nM T24983 CUIQ94 10014924 Ki = 32 nM T24983 C5ZJ4W 10015731 Ki = 17.6 nM T24983 CFM38B 10017758 Ki = 28 nM T24983 CA80TJ 10018402 EC50 = 3150 nM T24983 CTK42D 10018480 Ki = 60 nM T24983 CHP51K 10020098 EC50 = 52 nM T24983 C1VDL8 10021193 Ki = 3 nM T24983 CXBN42 10021692 Ki = 1300 nM T24983 C12TXY 10022369 EC50 = 159 nM T24983 CL6D7O 10023466 Ki = 4.3 nM T24983 C84EIF 10024158 EC50 = 66 nM T24983 C3MK8V 10039198 Ki = 54 nM T24983 CGTA58 10040546 Ki = 400 nM T24983 C1MJV4 10041417 Ki = 22 nM T24983 CORP02 10042205 EC50 = 270 nM T24983 CM12SD 10042826 EC50 = 346 nM T24983 CN1M6G 10042972 Ki = 2.4 nM T24983 C0HVU6 10044835 Ki = 4 nM T24983 CJI9F1 10045314 EC50 = 160 nM T24983 CFXD46 10045525 Ki = 4 nM T24983 C8WPO6 10049549 Ki = 5.012 nM T24983 CX27EK 10049758 IC50 = 570 nM T24983 C4GHO2 10053476 Ki = 150 nM T24983 CLNY93 10058787 Ki = 269 nM T24983 C6Y3NO 10063875 Ki = 359 nM T24983 CLW45Q 10064956 EC50 = 512 nM T24983 CQ2CS1 10064981 Ki = 14.8 nM T24983 C4PCO3 10065083 Ki = 6.53 nM T24983 CT2OG9 10065188 Ki = 32 nM T24983 CT5VE4 10066168 EC50 = 62 nM T24983 C8Z6MA 10067306 IC50 > 5000 nM T24983 CO69FB 10069973 Ki = 3.94 nM T24983 C4LQY1 10071413 Ki = 23.99 nM T24983 C5HJ1G 10073022 Ki = 68.1 nM T24983 C03KWH 10073194 Ki = 28 nM T24983 CJ16VZ 10084583 Ki = 50 nM T24983 CB8K0C 10086123 Ki = 330 nM T24983 CX6L2Q 10086348 Ki = 371 nM T24983 CGW9L7 10088259 EC50 = 1.2 nM T24983 C0D4UB 10088811 EC50 = 50 nM T24983 C6BDZ3 10089203 Ki = 250 nM T24983 C7O8VH 10092041 IC50 = 280 nM T24983 CJXQ40 10092819 Ki = 30 nM T24983 CA3LE2 10098342 Ki = 3090.3 nM T24983 C54EYD 10108561 IC50 = 251.19 nM T24983 CKCI50 10110263 Ki = 96 nM T24983 C0HAD8 10115074 Ki = 29 nM T24983 CL7N8S 10131111 Ki = 22 nM T24983 COXA05 10133031 Ki = 5.3 nM T24983 CWT32F 10137747 Ki = 65 nM T24983 C8X4BP 10137748 Ki = 34 nM T24983 C5JZ9P 10157556 Ki = 3 nM T24983 CR62CZ 10158455 Ki = 9 nM T24983 C1DQ8L 10161526 Ki = 2145 nM T24983 CB30TC 10176799 Ki = 26 nM T24983 C2ZC0Q 10183626 Ki = 1346 nM T24983 CZ97UO 10184153 Ki = 603 nM T24983 CZKG96 10200496 Ki = 14.1 nM T24983 CMJ2W9 10220333 Ki = 3 nM T24983 CWR4J6 10220541 Ki > 3330 nM T24983 CY2S4Z 10224165 Ki = 19 nM T24983 C2YZG0 10225902 EC50 = 416 nM T24983 CGJ5Q9 10225942 Ki = 2243 nM T24983 CS3X6I 10229397 Ki = 2438 nM T24983 CO64WJ 10236758 Ki = 0.9772 nM T24983 COZ2S7 10242548 Ki = 485 nM T24983 CYCQ58 10245409 Ki = 2 nM T24983 CVF1E5 10246054 IC50 > 1000 nM T24983 CFCP96 10247720 Ki = 0.95 nM T24983 CY82IS 10248715 Ki = 0.96 nM T24983 CW8O2L 10249308 Ki = 2.8 nM T24983 CWD35Q 10249755 Ki = 6.31 nM T24983 CC1PJ7 10251080 Ki = 12 nM T24983 COB28U 10254390 Ki = 720 nM T24983 CM5IJ7 10268039 EC50 = 100 nM T24983 CE9Y8J 10276451 Ki = 170 nM T24983 C9MPY2 10300403 Ki = 2314 nM T24983 C0L8VZ 10301202 Ki = 1118 nM T24983 C8XKC0 10310103 Ki = 7000 nM T24983 CT91NH 10314506 EC50 = 85 nM T24983 CJ3Q1T 10314824 Ki = 1 nM T24983 C5R8TC 10315310 Ki = 0.5248 nM T24983 C78YSD 10316440 EC50 = 126 nM T24983 CB8O9X 10318141 Ki = 8.2 nM T24983 CHJ4W9 10335148 Ki = 34 nM T24983 C9P6BG 10335627 EC50 = 532 nM T24983 CLS0X1 10336039 Ki = 1.6 nM T24983 CC3Z4E 10338536 EC50 = 2460 nM T24983 C4RQX5 10339711 EC50 = 180 nM T24983 CYP68J 10356955 Ki = 9.5 nM T24983 C4A0PF 10357628 Ki = 26 nM T24983 C1RX9F 10357631 Ki = 275.42 nM T24983 CQ08TM 10359019 EC50 = 1 nM T24983 C1NTD8 10359539 Ki = 310 nM T24983 CTY10B 10359645 EC50 = 840 nM T24983 CDCX49 10359736 Ki = 7.943 nM T24983 CXAK13 10359942 Ki = 1.3 nM T24983 C32KOP 10360923 Ki = 5.2 nM T24983 CD4H6R 10361512 Ki = 2.3 nM T24983 C8LT7J 10363821 Ki = 109 nM T24983 CH1IY6 10375676 Ki = 76 nM T24983 CIX51R 10378194 EC50 = 1.9 nM T24983 CR3KU9 10380133 IC50 > 5000 nM T24983 CDAC63 10381889 IC50 = 2.63 nM T24983 C6DFI4 10382581 Ki = 6.7 nM T24983 CKG4U7 10383571 EC50 = 685 nM T24983 CI5QO8 10383724 EC50 = 100 nM T24983 C9DJY1 10385089 EC50 = 45 nM T24983 CH2SF5 10385883 EC50 = 85 nM T24983 CLY48W 10385977 Ki = 37 nM T24983 C4DZ0M 10392655 Ki = 800 nM T24983 C6J2ZL 10402378 Ki = 546 nM T24983 CJNR48 10403092 Ki = 54 nM T24983 CT07SM 10403435 Ki = 37 nM T24983 CX2Y7J 10403608 Ki = 1 nM T24983 C4OF7Y 10404663 Ki = 3000 nM T24983 CQ1B2S 10404821 EC50 = 68 nM T24983 CN3PQ7 10404935 EC50 = 38 nM T24983 C82MVD 10405922 EC50 = 340 nM T24983 CP8N0D 10405923 EC50 = 324 nM T24983 C94PNM 10406796 IC50 = 1 nM T24983 C04WGF 10407367 IC50 > 5000 nM T24983 C9R6GC 10411988 Ki = 117 nM T24983 CH5M7W 10413085 Ki = 15.85 nM T24983 CGTF70 10424172 Ki = 12 nM T24983 C2SLJ9 10424961 Ki = 320 nM T24983 CZ5HC6 10425024 Ki = 228 nM T24983 CO76HW 10425969 Ki = 3.9 nM T24983 CA3PI9 10427977 Ki = 1.2 nM T24983 CB53UA 10428669 EC50 = 115 nM T24983 CH6DK1 10428816 EC50 = 63 nM T24983 CA1FD2 10430685 Ki = 318 nM T24983 CN6IG8 10430781 EC50 = 135 nM T24983 CD86MZ 10430816 Ki = 63.6 nM T24983 CL0ZB2 10430935 Ki = 28.1 nM T24983 C8ZA3G 10432808 Ki = 46 nM T24983 C9A4MJ 10436285 Ki = 1116 nM T24983 C4UN0A 10436653 Ki = 35 nM T24983 C8KD1B 10438027 Ki = 1720 nM T24983 C1CO4G 10447709 Ki = 0.955 nM T24983 CPN63D 10449136 Ki = 150 nM T24983 CG95BJ 10449865 EC50 = 90 nM T24983 CL8HQ6 10450082 IC50 = 20 nM T24983 C47IOH 10450375 Ki = 0.7 nM T24983 CVPK09 10450880 Ki = 8.7 nM T24983 C1SZU3 10450892 Ki = 0.52 nM T24983 CW0ND4 10454026 Ki = 476 nM T24983 C04MGE 10454684 Ki = 3 nM T24983 C05PSB 10456166 Ki > 800 nM T24983 CK57FH 10469437 Ki = 29 nM T24983 CV9N7G 10470579 Ki = 313 nM T24983 COV85C 10472143 Ki = 36 nM T24983 C5LBS7 10472158 IC50 > 5000 nM T24983 C24UJV 10472323 EC50 = 420 nM T24983 CUW3M2 10473658 Ki = 3.467 nM T24983 C7HI4X 10474613 Ki = 26 nM T24983 CPI5M7 10476504 Ki = 2 nM T24983 CE79QV 10477871 Ki = 39.81 nM T24983 CEF2O6 10478367 Ki > 10000 nM T24983 CFLZ47 10479188 Ki = 11 nM T24983 CEP10Q 10479822 Ki = 630.96 nM T24983 CD3A2O 10492351 Ki > 2500 nM T24983 C2WNH9 10494394 Ki = 1.2 nM T24983 C4JWB8 10494689 Ki = 73 nM T24983 CEY43J 10495652 Ki = 9 nM T24983 CP51BI 10495881 Ki = 73 nM T24983 CQB58X 10496095 IC50 = 73 nM T24983 C3ZW8P 10497179 Ki = 19 nM T24983 C7VC6L 10497193 Ki = 110 nM T24983 CQ72YM 10497674 IC50 = 10 nM T24983 CX1UD7 10498094 Ki = 1.4 nM T24983 CHUF43 10498196 Ki = 6.7 nM T24983 CRUT74 10498972 Ki = 26.92 nM T24983 C31HYJ 10501113 IC50 = 7.8 nM T24983 CN9BT6 10512444 Ki = 1033 nM T24983 CN28AB 10515841 Ki = 193 nM T24983 C1GRL4 10518406 Ki = 5.37 nM T24983 C01NJM 10519543 Ki = 4.4 nM T24983 C49BOW 10520781 Ki = 420 nM T24983 CYL86S 10520941 Ki = 10 nM T24983 C8ZMA1 10522334 Ki = 930 nM T24983 C12ZTU 10522613 Ki = 0.56 nM T24983 C38ACZ 10522614 Ki = 0.86 nM T24983 C3EG1O 10524285 Ki = 199.53 nM T24983 C7TZ3K 10524751 Ki = 1400 nM T24983 CQ5F3N 10525119 Ki = 5.012 nM T24983 CB7OK1 10541769 IC50 > 10000 nM T24983 C9ZYA3 10542345 Ki = 30 nM T24983 CRF7P9 10543298 Ki = 4 nM T24983 C12SBD 10543353 Ki > 1000 nM T24983 C59NSH 10543696 Ki = 1400 nM T24983 C27FUN 10544707 Ki = 63 nM T24983 C8ZG3C 10545941 Ki = 3.8 nM T24983 CXI49Z 10546453 Ki = 5.5 nM T24983 C7UCS1 10546540 Ki = 0.33 nM T24983 C40CJM 10546828 Ki = 47 nM T24983 CYF64N 10547607 Ki = 0.64 nM T24983 C23BRU 10548105 Ki = 38 nM T24983 CKD0F6 10548329 Ki = 19.95 nM T24983 CQ2R5D 10548967 Ki = 141 nM T24983 C4VZ2K 10549355 Ki = 4.7 nM T24983 CQD6C8 10551026 Ki = 5 nM T24983 CH7E0W 10559624 Ki = 729 nM T24983 CJH5T9 10567430 Ki = 3.6 nM T24983 CBP4X5 10567507 Ki = 4 nM T24983 C08LPE 10567839 Ki = 74 nM T24983 C0HJS2 10568183 IC50 = 85 nM T24983 CWG62F 10568740 Ki = 2700 nM T24983 CC56ON 10568805 Ki = 7.9 nM T24983 CYL67U 10569690 Ki = 71 nM T24983 C60SMR 10570080 Ki = 2 nM T24983 C7YM3R 10570479 Ki = 1.1 nM T24983 CW38OC 10570563 Ki = 6 nM T24983 C6S0TG 10570898 Ki = 7.5 nM T24983 C1YU3Q 10571927 Ki = 2.1 nM T24983 CZ6XT2 10572229 Ki = 201 nM T24983 CZ87BA 10572985 Ki = 391 nM T24983 CM3C1L 10573099 Ki = 280 nM T24983 C02HSA 10574303 Ki = 4.5 nM T24983 C0S3AJ 10574818 Ki = 3.3 nM T24983 C9SP3R 10587140 Ki = 470 nM T24983 COL98E 10588194 Ki = 1.995 nM T24983 CP1Y7K 10589218 Ki = 2.692 nM T24983 CT2R7G 10589834 IC50 > 10000 nM T24983 C12ZRK 10590285 Ki = 10.96 nM T24983 CRJ13B 10593191 Ki = 3.388 nM T24983 C8E4HR 10593869 Ki = 4.5 nM T24983 C97NMI 10594054 Ki = 3.4 nM T24983 CM7Z9X 10594113 Ki = 9.1 nM T24983 C17ZDI 10594242 Ki = 1 nM T24983 CTZ9V3 10594723 IC50 = 133 nM T24983 CD27FZ 10594764 Ki = 0.75 nM T24983 C1VLS4 10595646 Ki = 25.12 nM T24983 CDO93P 10595908 Ki = 1.5 nM T24983 C57DKO 10596380 IC50 > 1000 nM T24983 C9S0RY 10597050 Ki = 416 nM T24983 CK9LD1 10597114 Ki = 492 nM T24983 C7GDX0 10612157 Ki = 16.6 nM T24983 CH49UB 10613605 Ki = 2174 nM T24983 C3FS5U 10615437 Ki = 11 nM T24983 CSI97L 10615684 IC50 = 8 nM T24983 C9JI3A 10615787 Ki = 1.4 nM T24983 CB6HW4 10615990 IC50 = 68 nM T24983 C5XI7L 10616050 Ki = 21.88 nM T24983 CPY43H 10617133 IC50 = 6 nM T24983 C56UGP 10617366 Ki = 3.1 nM T24983 CT5A6H 10617381 Ki = 12 nM T24983 CWQ76V 10617946 Ki = 410 nM T24983 C6QB8L 10618211 Ki = 12 nM T24983 C2LN0J 10618874 Ki = 5.5 nM T24983 CJ7R5F 10618875 Ki = 1.6 nM T24983 C3VQK1 10619612 Ki = 12 nM T24983 CJ40ZT 10619737 Ki = 1.2 nM T24983 CDZ16W 10620139 Ki = 8.5 nM T24983 CG0MN7 10623982 Ki = 87 nM T24983 C6HAV3 10636896 Ki = 74 nM T24983 CKF8L2 10637198 IC50 > 10000 nM T24983 C0V5NM 10638052 Ki = 0.8 nM T24983 CJON98 10639353 Ki = 19 nM T24983 C8O4BC 10639430 Ki = 50 nM T24983 C9D5MP 10640530 Ki = 2.6 nM T24983 CK4O3W 10641637 Ki = 29 nM T24983 C2B5NL 10641783 Ki = 5 nM T24983 C89NYU 10641954 Ki = 34 nM T24983 C0DCY3 10641955 Ki = 17 nM T24983 CKP3A1 10642106 Ki = 62.4 nM T24983 CPTF56 10642239 EC50 = 15 nM T24983 COX0D5 10642702 Ki = 325 nM T24983 CED15G 10643588 Ki = 0.71 nM T24983 CL8KB3 10643589 Ki = 5.2 nM T24983 CD21IV 10643697 Ki = 1.8 nM T24983 C4K0PA 10643780 Ki = 9 nM T24983 C6TZS3 10644771 Ki = 25 nM T24983 C5EQ1V 10646459 Ki = 2.7 nM T24983 C3VMO5 10646834 Ki = 7 nM T24983 C2W5BE 10660814 Ki = 0.4571 nM T24983 C15GLS 10662508 Ki > 3300 nM T24983 CFC38D 10663221 Ki = 50 nM T24983 CTP8L0 10664621 Ki = 2.6 nM T24983 C43FER 10665101 Ki = 15.85 nM T24983 CU3XJ4 10665598 Ki = 17 nM T24983 CI2OT7 10665626 Ki = 16 nM T24983 CCU12E 10666005 IC50 = 3 nM T24983 C31ZOC 10666315 Ki = 1.1 nM T24983 CWE53T 10667201 Ki = 5.5 nM T24983 C7K9DP 10667579 Ki = 0.46 nM T24983 C4IY3Z 10667966 Ki = 1900 nM T24983 CT45YR 10668173 IC50 = 45 nM T24983 C8C3QP 10669042 Ki = 0.67 nM T24983 CU31PH 10682854 Ki = 1504 nM T24983 CO49AQ 10683127 Ki > 3300 nM T24983 CZLJ52 10684706 Ki = 3.09 nM T24983 C0ZCG1 10684789 Ki = 570 nM T24983 C6R7JD 10685891 Ki = 8.7 nM T24983 CJGP65 10687228 Ki > 3300 nM T24983 C7T2FU 10687362 Ki = 7.5 nM T24983 CY4Z1R 10687967 Ki = 160 nM T24983 CBW96O 10688035 Ki = 22 nM T24983 C60DRH 10688036 Ki = 23 nM T24983 C8QVK3 10688157 Ki = 74 nM T24983 C87BLK 10688561 IC50 = 31 nM T24983 CJFP08 10688858 IC50 = 29 nM T24983 CK0TC9 10688859 IC50 = 30 nM T24983 CMVD23 10689266 Ki = 84 nM T24983 CC1E7W 10690200 Ki = 1.7 nM T24983 C75DXM 10690882 Ki = 19.95 nM T24983 CEM56L 10691523 Ki = 20 nM T24983 CD1KF8 10691599 Ki = 3.6 nM T24983 CR2FI0 10691634 Ki = 31.62 nM T24983 CHZ8O2 10692886 Ki = 212 nM T24983 CEVQ74 10693793 Ki = 5.6 nM T24983 C8OC6U 10704110 Ki = 32 nM T24983 CU25LW 10708280 Ki = 0.52 nM T24983 CSXO03 10713599 IC50 = 164 nM T24983 CE5QA3 10713620 Ki = 68 nM T24983 C4O6KG 10714184 Ki = 350 nM T24983 CIQ45P 10715225 Ki = 21 nM T24983 CA8MK0 10715375 Ki = 5.012 nM T24983 C7TPN8 10716772 Ki = 1.5 nM T24983 CT7Y9K 10716980 Ki = 2.1 nM T24983 CK04WL 10719212 Ki = 4.4 nM T24983 C71VBX 10732925 Ki = 1.096 nM T24983 CWY6V1 10733406 Ki = 0.309 nM T24983 CO9BL7 10734727 Ki = 0.8318 nM T24983 CHN4A3 10735344 Ki = 23 nM T24983 CQ2DU0 10735405 Ki = 18 nM T24983 CO1DT0 10735463 Ki = 6 nM T24983 CJM1R5 10737150 Ki = 204 nM T24983 CNWC38 10737474 Ki = 5.248 nM T24983 CY5HG9 10738530 Ki = 110 nM T24983 C65DWL 10739194 IC50 = 16 nM T24983 CMXR17 10740483 Ki = 1.3 nM T24983 C4RAC7 10740968 Ki = 22 nM T24983 C61BCK 10740969 Ki = 67 nM T24983 CLM1O5 10741841 Ki = 3.4 nM T24983 C9Z8TB 10757990 Ki > 7300 nM T24983 C8XD2C 10758004 Ki = 5.6 nM T24983 C19UPY 10759511 Ki = 4.3 nM T24983 C21TFA 10759963 Ki > 10000 nM T24983 CH5AY1 10760638 Ki = 3.89 nM T24983 CHN8T2 10760813 Ki = 13 nM T24983 C9FE7Z 10761040 IC50 = 9 nM T24983 CDNE69 10761258 Ki = 40.74 nM T24983 CF06YO 10761828 Ki = 646 nM T24983 CAV6N0 10761912 Ki = 42 nM T24983 CC2L1A 10762432 Ki = 1.3 nM T24983 C80STM 10763496 Ki = 46 nM T24983 CQ2R0A 10780076 IC50 = 96 nM T24983 C3LB9N 10780510 Ki = 0.3467 nM T24983 CU9T8V 10780942 Ki = 4.365 nM T24983 C2QJP8 10781960 Ki = 30 nM T24983 C2MPX6 10782049 Ki = 33 nM T24983 CT8F3Y 10782097 Ki = 2664 nM T24983 CIDM49 10782111 IC50 = 37 nM T24983 C5N3RM 10782946 Ki = 11 nM T24983 C6D3BX 10783358 Ki = 0.63 nM T24983 C4G8HB 10783874 Ki = 0.84 nM T24983 C6J2FC 10786367 Ki = 60 nM T24983 CF9S6Q 10786474 Ki = 180 nM T24983 CCBO47 10786591 Ki = 61 nM T24983 C2GO7R 10790517 Ki = 110 nM T24983 CXO6J4 10801405 Ki = 335 nM T24983 CL1CV6 10801925 Ki = 256 nM T24983 C46LYA 10803754 IC50 = 567 nM T24983 CP74YO 10803828 Ki = 529 nM T24983 CB74KW 10803829 Ki = 292 nM T24983 CB45KG 10805355 Ki = 4.365 nM T24983 CF1LE7 10805797 Ki = 410 nM T24983 C5M9AW 10806501 Ki = 52 nM T24983 CNWV56 10807035 Ki = 11 nM T24983 CS7YU8 10807795 Ki = 2.6 nM T24983 CRZU91 10808230 IC50 = 9 nM T24983 C24QAM 10809899 Ki = 1.1 nM T24983 CS0BT5 10810976 Ki = 42 nM T24983 C1VTJ3 10811814 Ki = 241 nM T24983 CZ1F3B 10824155 Ki = 3900 nM T24983 C1SK9V 10826290 Ki = 1200 nM T24983 CJ9BY0 10827222 Ki = 676.08 nM T24983 CE7M9P 10829708 IC50 = 3 nM T24983 CCN52S 10830557 Ki = 110 nM T24983 CC9S2I 10830804 Ki = 2200 nM T24983 C1QMR4 10831735 Ki = 2.1 nM T24983 CJ1DI4 10831786 Ki = 4800 nM T24983 CL4T8O 10832341 Ki = 23 nM T24983 C4R7DC 10832895 IC50 = 4 nM T24983 CM83SE 10833953 Ki = 7.5 nM T24983 CRZ3T2 10836365 Ki = 3 nM T24983 C4IFV1 10837488 Ki = 1.9 nM T24983 CQ29GV 10837493 Ki = 20 nM T24983 CC8ZP3 10837494 Ki = 18 nM T24983 C14VQN 10851217 IC50 = 48 nM T24983 CF1S7E 10852461 Ki = 150 nM T24983 CL8Q9F 10854185 Ki = 16 nM T24983 CPU26G 10854370 Ki = 2.8 nM T24983 C53OXZ 10861560 Ki = 22.3 nM T24983 C9A8KN 10862425 Ki = 40 nM T24983 CZYF05 10871118 Ki = 64 nM T24983 C1UQ4H 10873318 Ki = 55 nM T24983 CKOF21 10873956 Ki > 800 nM T24983 CMV36C 10884046 Ki = 44 nM T24983 CD3U9P 10885524 Ki = 391 nM T24983 CRI50E 10885636 IC50 = 776 nM T24983 CL4S8G 10893228 Ki = 163 nM T24983 CB1HY3 10894144 IC50 = 1410 nM T24983 C1GW5K 10894276 Ki = 183 nM T24983 CU80EA 10895106 Ki = 77.62 nM T24983 CWJL70 10905740 IC50 = 6550 nM T24983 C8CZB9 10905940 Ki = 7.3 nM T24983 CS7GO8 10906255 Ki > 1000 nM T24983 CL8AG5 10917920 Ki = 3000 nM T24983 C2UZ8H 10917953 Ki = 5700 nM T24983 C6D7JR 10924369 Ki = 160 nM T24983 CNT3E2 10926404 Ki = 11 nM T24983 C67FYJ 10927750 Ki = 679 nM T24983 CGZA42 10939167 Ki = 27 nM T24983 C0UGV5 10939222 Ki = 50.12 nM T24983 C69ULE 10939408 Ki = 370 nM T24983 CC07JE 10942784 Ki > 3333 nM T24983 CNB39C 10947658 Ki = 18 nM T24983 CN7XS4 10948527 IC50 = 947 nM T24983 CO7P5V 10948748 Ki = 0.04 nM T24983 C0WX2Y 10950176 Ki = 9 nM T24983 C3JCI2 10960333 Ki = 6800 nM T24983 CH14OY 10961938 Ki = 720 nM T24983 C9HPJ3 10972865 Ki = 350 nM T24983 C5NRU3 10973768 Ki = 3600 nM T24983 CFU1S9 10980338 Ki = 3.1 nM T24983 C2HP7F 10981761 IC50 = 1880 nM T24983 CB86ST 10983150 Ki = 105 nM T24983 CWQ40B 10994141 Ki = 604 nM T24983 C0FV9Z 11003833 Ki = 3.1 nM T24983 CJC9K4 11005810 IC50 = 543 nM T24983 CO36VS 11005852 Ki = 530 nM T24983 CXZ29Y 11016342 Ki = 283 nM T24983 CH9GU5 11016418 Ki = 4900 nM T24983 CT56RB 11026289 Ki = 1380 nM T24983 CQ6M1S 11028157 Ki = 652 nM T24983 C4Y9XK 11033734 Ki = 47 nM T24983 CB7N1P 11035765 IC50 = 429 nM T24983 CJ15OI 11036114 Ki = 0.26 nM T24983 C01NDT 11036640 Ki = 40.74 nM T24983 CU6HR7 11036641 Ki = 14 nM T24983 CC1YO2 11049209 Ki = 6400 nM T24983 C0SUF4 11057969 Ki = 0.67 nM T24983 CNBO86 11058535 Ki > 1000 nM T24983 CT9CZ1 11058829 Ki = 40 nM T24983 CE3J0B 11068912 Ki = 30 nM T24983 CAO5X2 11070520 Ki > 1000 nM T24983 CG41BK 11071079 IC50 = 338 nM T24983 CUJ4W7 11071135 Ki = 7200 nM T24983 CG63OS 11077918 Ki = 1300 nM T24983 CNF43K 11078813 Ki = 3600 nM T24983 CE85YF 11079832 Ki = 37 nM T24983 C9LCB6 11090403 Ki = 0.21 nM T24983 CM2BD4 11092112 Ki = 7500 nM T24983 C7DE0U 11113605 IC50 = 716 nM T24983 CVE8T3 11121216 Ki = 72 nM T24983 CVM23D 11123162 Ki > 800 nM T24983 C8TW2P 11131951 Ki = 0.025 nM T24983 CE8FH4 11132372 Ki > 1000 nM T24983 CTXS48 11133385 Ki = 2170 nM T24983 CWG8O0 11133533 Ki = 168 nM T24983 CXP12A 11133602 Ki = 67.61 nM T24983 CWT4S5 11144835 Ki = 345 nM T24983 CHD24Z 11151081 EC50 = 39.2 nM T24983 CW5ER6 11151135 Ki = 850 nM T24983 C9MWB5 11151919 EC50 = 45 nM T24983 CEX52K 11151920 Ki = 32.1 nM T24983 CU08BT 11152225 Ki = 920 nM T24983 CMTB75 11153076 Ki = 4.9 nM T24983 C3Q9UG 11154178 Ki > 10000 nM T24983 CZ0KA8 11156017 Ki = 24 nM T24983 CNE31P 11163137 EC50 = 24.1 nM T24983 C4K6QP 11164276 EC50 = 37.2 nM T24983 CZ2F5M 11164922 Ki = 61 nM T24983 CQ7ZA0 11175610 EC50 = 164 nM T24983 C42PWL 11176211 Ki = 35 nM T24983 CN06GJ 11186895 Ki > 1000 nM T24983 CBE97D 11187628 Ki = 61 nM T24983 C3CIH1 11187957 EC50 = 46.4 nM T24983 C7UL1W 11197141 Ki > 10000 nM T24983 CG7D2K 11198974 EC50 = 320 nM T24983 C8PF9M 11199162 EC50 = 37.6 nM T24983 C4CW6X 11200205 Ki = 6.4 nM T24983 C9N5QU 11200511 Ki > 5000 nM T24983 CI0M3S 11211058 EC50 = 46 nM T24983 CXO67U 11213037 Ki = 239.88 nM T24983 C5XNA7 11220975 Ki = 26.5 nM T24983 C6V2QH 11221906 Ki = 27.5 nM T24983 CEFK20 11222637 EC50 = 95 nM T24983 C6D1MZ 11223004 Ki > 5000 nM T24983 C8RJ3D 11223303 Ki > 10000 nM T24983 C6LB4S 11230330 Ki = 40 nM T24983 CET64Y 11233944 Ki = 5.4 nM T24983 CKX06B 11235174 Ki > 10000 nM T24983 C7N5FP 11245414 Ki = 100 nM T24983 C18ORY 11255258 EC50 = 23 nM T24983 CL04EZ 11256262 EC50 = 28.5 nM T24983 CH92LP 11256583 EC50 = 63.7 nM T24983 CM72YX 11269330 Ki = 5060 nM T24983 CD47FC 11269392 EC50 = 249 nM T24983 CKN4L3 11280225 EC50 = 135 nM T24983 CUJ2R7 11280344 Ki = 22.5 nM T24983 C1GO5D 11280787 Ki = 52 nM T24983 CZY6I5 11290928 Ki = 29 nM T24983 C8LAP9 11292299 EC50 = 296 nM T24983 CJ9N6I 11292776 Ki = 9.3 nM T24983 CC2Y4X 11299620 Ki = 47 nM T24983 CRZX70 11300847 Ki = 376 nM T24983 C2ABW4 11301354 EC50 = 21.7 nM T24983 CH0X7A 11303390 Ki = 46 nM T24983 CQ2Z6J 11304676 Ki = 47.9 nM T24983 CCZ8S3 11314005 Ki = 83 nM T24983 CI56TH 11314352 EC50 = 56.6 nM T24983 CKDU17 11315028 Ki = 4.5 nM T24983 C9RW3C 11324794 Ki = 22.8 nM T24983 CIZH05 11325334 Ki = 14.2 nM T24983 CP5AF8 11325645 EC50 = 175 nM T24983 CF38AZ 11325818 EC50 = 113 nM T24983 CF0SE7 11328099 Ki = 430 nM T24983 CIK35D 11336814 Ki = 6.4 nM T24983 C4XME0 11338828 Ki = 7 nM T24983 C0NRE8 11346967 Ki > 10000 nM T24983 CSB26G 11347425 Ki = 79.6 nM T24983 CW75OZ 11348526 Ki = 180 nM T24983 CCY23Q 11351639 Ki = 1770 nM T24983 CA1NC6 11356479 Ki = 58 nM T24983 CXWH42 11358377 Ki > 10000 nM T24983 C1TNF0 11360382 Ki = 32 nM T24983 C26PKR 11360927 Ki = 1000 nM T24983 CCVK79 11370781 EC50 = 33.3 nM T24983 CBPJ98 11371795 EC50 = 42.3 nM T24983 CJ42PI 11372852 Ki = 2.9 nM T24983 CY24NV 11374299 Ki > 10000 nM T24983 C82QCU 11375068 Ki = 520 nM T24983 CQ3V4K 11382447 Ki = 70 nM T24983 C1PUI4 11383473 Ki = 32 nM T24983 CBV52J 11384146 Ki > 5000 nM T24983 C1OM3C 11384207 Ki = 281.84 nM T24983 C4SZ7W 11384664 Ki = 199.53 nM T24983 COY20M 11392147 EC50 = 11 nM T24983 CT0FG4 11393899 Ki = 32 nM T24983 CGJ2Z7 11394708 EC50 = 84 nM T24983 C1V4EQ 11404156 Ki > 10000 nM T24983 CDV4A0 11405107 Ki = 83 nM T24983 CR8T2W 11405182 Ki = 200 nM T24983 CT32OJ 11406143 Ki > 10000 nM T24983 COZJ34 11406804 Ki = 13 nM T24983 C2R1SC 11407122 Ki = 400 nM T24983 CGN10L 11408148 Ki = 1070 nM T24983 CJUI62 11416883 EC50 = 91 nM T24983 CVB47W 11417804 Ki = 40 nM T24983 CZ0TA2 11417962 Ki = 23 nM T24983 CIS2D5 11428005 Ki = 650 nM T24983 C8MY7G 11428416 Ki = 13 nM T24983 CO6F2D 11431895 Ki > 5000 nM T24983 CBN91Q 11439190 Ki = 10000 nM T24983 CY1M6Q 11450607 EC50 = 40.1 nM T24983 C86CJB 11451022 Ki = 4.5 nM T24983 CA3JG1 11451703 Ki = 71.2 nM T24983 C6SVK9 11452692 Ki = 804 nM T24983 CB3P6S 11452916 Ki > 10000 nM T24983 C05VEA 11453253 Ki = 169.82 nM T24983 CFTR78 11464857 Ki = 2 nM T24983 CTA58W 11469395 Ki > 33333 nM T24983 C8L6ZI 11472028 Ki > 10000 nM T24983 C4GTH7 11474021 Ki = 30 nM T24983 C3NVL1 11474209 EC50 = 136 nM T24983 CLZ91D 11474734 EC50 = 285 nM T24983 CK39HZ 11486421 Ki > 10000 nM T24983 CTU1Z7 11488247 Ki = 4331 nM T24983 CAL0Z7 11488451 Ki = 265 nM T24983 CN63TR 11504230 Ki = 5.4 nM T24983 C9BT2W 11512263 Ki = 288.4 nM T24983 C59SCV 11516033 Ki = 0.99 nM T24983 CAMP52 11517928 Ki = 120 nM T24983 CC6U7R 11522476 Ki = 2514 nM T24983 CO0R2G 11540842 Ki = 251.19 nM T24983 CN3W7S 11543350 Ki > 10000 nM T24983 C5ZY6N 11545813 Ki = 41.8 nM T24983 C7QKD5 11547151 Ki = 977.24 nM T24983 C7S2WZ 11558055 Ki = 11.3 nM T24983 C1V5CH 11559090 Ki > 10000 nM T24983 CY5I0U 11559581 Ki = 2 nM T24983 C9UH2M 11559589 Ki = 3 nM T24983 CH67TN 11560697 Ki = 840 nM T24983 C8GK0U 11566745 Ki = 165 nM T24983 C5J2UP 11569619 Ki = 281.84 nM T24983 CRK97Z 11570471 Ki = 75.86 nM T24983 C32JGN 11570589 Ki = 39.81 nM T24983 CTG5X1 11574902 Ki = 0.25 nM T24983 C8NMI4 11575479 Ki > 10000 nM T24983 C1Q8LC 11575799 Ki = 0.99 nM T24983 CE60FY 11576528 Ki = 158.49 nM T24983 C8CU1X 11581237 Ki = 1.6 nM T24983 C4BGF8 11581443 Ki = 170 nM T24983 CQ09NJ 11583188 Ki = 0.33 nM T24983 CI2FK6 11584858 Ki = 41.69 nM T24983 CU45DK 11595209 Ki > 10000 nM T24983 CZPE61 11608015 Ki > 3333 nM T24983 C9VOB8 11613105 Ki = 269.15 nM T24983 C9BZG0 11615489 Ki = 58 nM T24983 C62SOL 11615782 Ki = 16000 nM T24983 CR6S3I 11624518 Ki = 170 nM T24983 CC2G9I 11626748 Ki = 1900 nM T24983 C8R6MK 11630058 Ki = 90000 nM T24983 CS4CR7 11631304 Ki > 5000 nM T24983 C8ZU2X 11631892 Ki = 1.3 nM T24983 C7CZE3 11633170 Ki = 2.3 nM T24983 CMZR85 11633816 Ki = 257 nM T24983 CG1C3D 11637457 Ki = 99 nM T24983 C2OU7Y 11638332 Ki > 10000 nM T24983 CI17EA 11638780 Ki = 4 nM T24983 CEN25S 11646648 Ki = 567 nM T24983 C9XD0H 11649431 Ki = 218.78 nM T24983 CEZO71 11652518 Ki = 2800 nM T24983 C1HDM5 11653679 Ki = 6.6 nM T24983 C5T4UV 11655570 Ki = 0.53 nM T24983 CP21DV 11658914 Ki = 200 nM T24983 C7NHO6 11659604 Ki = 500 nM T24983 CD79UX 11661609 Ki = 0.99 nM T24983 CO2HB4 11663604 Ki = 128.82 nM T24983 CPR2S8 11668034 Ki = 5 nM T24983 CY0J2U 11670421 Ki = 281.84 nM T24983 CH8M9X 11673558 Ki > 20000 nM T24983 CY4B9F 11676195 Ki = 0.63 nM T24983 CMQX39 11676873 Ki = 425 nM T24983 CTK8R9 11678172 Ki = 33 nM T24983 CSQ4B1 11681599 Ki = 18.7 nM T24983 CVRW29 11682812 Ki = 1.6 nM T24983 CS1WO0 11689612 Ki = 0.94 nM T24983 C3LYZ6 11694483 Ki = 14000 nM T24983 C1W8NR 11696910 Ki = 1.3 nM T24983 C9ED1Y 11697270 Ki = 0.84 nM T24983 CB4H2O 11699469 Ki = 140 nM T24983 C2YE9V 11699516 Ki = 91.2 nM T24983 CJL61W 11706497 Ki = 120 nM T24983 C3EP0X 11708363 Ki = 13000 nM T24983 CZ7SJ2 11716449 Ki = 378.5 nM T24983 C7T1IL 11720119 Ki = 302 nM T24983 CGO56C 11720302 Ki = 18 nM T24983 CDRB57 11724450 Ki = 2.7 nM T24983 CCS8F5 11724853 Ki = 120 nM T24983 CXYQ40 11725531 Ki = 1.5 nM T24983 CNPU72 11725909 Ki = 10 nM T24983 CZLY39 11726130 Ki = 100 nM T24983 CRQ45H 11726532 Ki = 1.7 nM T24983 CF7EC5 11729231 Ki = 0.018 nM T24983 C7PVL8 11730467 IC50 = 280 nM T24983 CB8WF0 11732013 Ki = 48 nM T24983 C10AGT 11738728 IC50 = 1 nM T24983 CP7IM3 11738945 EC50 = 26 nM T24983 CB0T3F 11739255 Ki = 8 nM T24983 C5OR8S 11739823 EC50 = 606 nM T24983 CL0SP1 11742798 Ki = 19 nM T24983 CPG15O 11743399 IC50 > 1000 nM T24983 CYV02C 11747350 Ki = 1600 nM T24983 CW1ZF7 11750030 Ki = 40 nM T24983 C5EH3J 11761412 Ki = 43 nM T24983 CQX0T6 11762743 Ki = 3990 nM T24983 C0FM6J 11771801 EC50 = 43.8 nM T24983 CXS18C 11772112 Ki = 11.4 nM T24983 C1T7NR 11772242 EC50 = 13.6 nM T24983 CXB48Q 11772767 Ki = 13.5 nM T24983 CBI6Z0 11774041 EC50 = 82 nM T24983 CC4D0K 11774177 Ki = 5.5 nM T24983 C2CB1X 11774358 Ki = 250 nM T24983 CV91RG 11778580 Ki = 375 nM T24983 C0L1XD 11779642 Ki = 190 nM T24983 CX0A6O 11783703 Ki = 84 nM T24983 CFCX90 11784097 Ki > 1000 nM T24983 C3RAX7 11784937 Ki = 35600 nM T24983 CT8LD5 11792163 Ki = 1.8 nM T24983 CAQP08 11792373 Ki = 12.3 nM T24983 CE61JV 11793892 Ki = 31.62 nM T24983 CAGO51 11793971 IC50 = 43 nM T24983 CEW12K 11794570 Ki = 44 nM T24983 CH03TX 11797442 Ki = 5.2 nM T24983 CFX10P 11809415 Ki = 356 nM T24983 C19GOZ 11811640 Ki = 7.58 nM T24983 CV68SD 11811808 Ki = 2.3 nM T24983 CWI40V 11811924 Ki > 1000 nM T24983 CWMA41 11812065 Ki = 368 nM T24983 CGFW41 11812838 Ki = 1140 nM T24983 CLR2Z9 11849181 Ki = 346 nM T24983 CLV61Z 11849182 Ki = 120 nM T24983 C0GM2D 11849184 EC50 = 4760 nM T24983 CL7YR2 11849225 EC50 = 17.5 nM T24983 C37OPA 11849228 EC50 = 382 nM T24983 CXG0L9 11849229 EC50 = 33 nM T24983 C1HSM3 11849262 EC50 = 109 nM T24983 CE83FP 11849263 EC50 = 2680 nM T24983 C5P7MQ 11849265 EC50 = 253 nM T24983 C8X2RG 11849266 Ki = 11.6 nM T24983 CPXD54 11849267 Ki = 67.1 nM T24983 CPEZ08 11849268 Ki = 90 nM T24983 C9YEI0 11849298 EC50 = 5370 nM T24983 C78XQP 11849299 EC50 = 3210 nM T24983 CN8ST9 11849634 EC50 = 25 nM T24983 CK80NX 11849635 EC50 = 20.3 nM T24983 CFM1V9 11849684 EC50 = 350 nM T24983 CKX4N9 11849729 EC50 = 48.7 nM T24983 C0MNQ3 11849730 EC50 = 338 nM T24983 CIG45B 11849731 EC50 > 10000 nM T24983 CD8B5E 11849734 EC50 = 139 nM T24983 CJ5Y2T 11849735 EC50 = 615 nM T24983 CEC2G8 11849736 EC50 = 81.8 nM T24983 CO9E3X 11849774 EC50 = 57.2 nM T24983 CU69CQ 11849775 Ki = 13.9 nM T24983 CXVA42 11849776 Ki = 20.1 nM T24983 CF6LX9 11849777 EC50 = 183 nM T24983 C3URG4 11849778 Ki = 6.3 nM T24983 CY06BF 11849779 EC50 = 74.7 nM T24983 CXA89H 11849780 EC50 = 341 nM T24983 CG1H7P 11849781 EC50 = 99 nM T24983 CZAX25 11849816 Ki = 134 nM T24983 C0XL3F 11849817 EC50 = 4290 nM T24983 C3D2KU 11849818 EC50 = 9.5 nM T24983 CJ0N9Z 11849819 EC50 = 41.7 nM T24983 CXY37C 11849820 EC50 = 33.5 nM T24983 CD8BQ7 11849821 EC50 = 22.6 nM T24983 COWM39 11849822 EC50 = 195 nM T24983 C4R6EA 11849823 EC50 = 44.8 nM T24983 CXLW54 11948707 Ki > 10000 nM T24983 CPKV28 11957618 Ki = 0.43 nM T24983 C7RY5S 11983282 Ki = 0.59 nM T24983 C02JVQ 12049520 Ki = 250 nM T24983 CXTH25 12049521 Ki = 370 nM T24983 C57VXR 12050193 Ki = 590 nM T24983 CV56XD 12050194 Ki = 1450 nM T24983 C5C2GB 12050195 Ki = 710 nM T24983 C64JUP 12050196 Ki = 590 nM T24983 C4QHA5 12050197 Ki = 370 nM T24983 CAL98J 12050198 Ki = 350 nM T24983 CJ7W9T 12050199 Ki = 390 nM T24983 CXEV76 12050200 Ki = 53 nM T24983 CP5W7X 12050201 Ki = 400 nM T24983 CZHQ31 12050202 Ki = 39 nM T24983 CX47WZ 12052258 Ki = 3.1 nM T24983 C6QEW2 12066264 Ki = 120 nM T24983 CF4D5H 12066265 Ki = 349 nM T24983 C9G7LR 12071089 Ki = 222 nM T24983 CT8SE7 12280575 Ki = 634 nM T24983 CHQ45V 12280580 Ki = 182 nM T24983 C4NWX9 12301195 Ki > 10000 nM T24983 CS3JE5 12581154 Ki = 603 nM T24983 C9XLS6 12581156 Ki = 1519 nM T24983 C72ZLP 12581164 Ki > 3333 nM T24983 CU3XH9 12581203 Ki = 964 nM T24983 CEBK96 12581219 Ki = 734 nM T24983 C5IVW7 12765116 Ki = 0.9 nM T24983 C28QEX 12765746 Ki = 1.5 nM T24983 CZT58X 12888943 Ki = 8.3 nM T24983 C8ON5D 12899499 Ki = 38.5 nM T24983 CPY6L8 12899569 Ki = 52.7 nM T24983 C5MB7I 12997400 Ki = 100 nM T24983 CXM15G 12997412 Ki = 791 nM T24983 CP0MN1 12997413 Ki = 326 nM T24983 C9C2UY 13014680 Ki = 2900 nM T24983 C1S2LW 13014681 Ki = 2700 nM T24983 CG7T8B 13014683 Ki = 1000 nM T24983 CHI9P5 13014692 Ki = 1 nM T24983 C2V9FL 13091268 Ki = 5.3 nM T24983 C2VAE5 13091273 Ki = 19.1 nM T24983 CC74ND 13373172 Ki = 5092 nM T24983 C68HWL 13457126 Ki = 60 nM T24983 CWS14H 13869641 Ki = 2.5 nM T24983 CSM29P 14665503 Ki = 210 nM T24983 CMO81H 14925759 EC50 = 0.1585 nM T24983 C5W4MG 15034333 Ki = 277 nM T24983 C5NVR4 15290395 Ki = 32 nM T24983 C4KNM7 15467369 Ki = 9.3 nM T24983 C5UO3R 15467370 Ki = 11 nM T24983 CCB94N 15467371 Ki = 5.7 nM T24983 C2B0NM 15467372 Ki = 160 nM T24983 CCMQ75 15467373 Ki = 125 nM T24983 C5FWQ2 15508238 Ki = 3300 nM T24983 C8VB3H 15508239 Ki = 2700 nM T24983 C5NC6J 15508242 Ki = 960 nM T24983 C72ERV 15512070 Ki = 2.8 nM T24983 C30CHU 15512229 Ki < 316.23 nM T24983 C15PZT 15522515 Ki = 17 nM T24983 CW50JX 15651970 Ki > 3333 nM T24983 CK5P6M 15651971 Ki > 3333 nM T24983 C59WZE 15654433 Ki > 933 nM T24983 C12WNY 15654434 Ki > 933 nM T24983 CT94FI 15817410 Ki = 3.5 nM T24983 CD30XV 15840855 IC50 = 7 nM T24983 C0UIX5 15840856 Ki = 8 nM T24983 CW9M5X 15888352 Ki = 78.6 nM T24983 C8UO1X 15981509 EC50 = 95 nM T24983 C0G2EO 16007117 Ki = 870 nM T24983 CWMC70 16090814 Ki = 98.4 nM T24983 CP09RQ 16090821 Ki = 184 nM T24983 CO0IQ4 16094665 EC50 = 9.8 nM T24983 C5Q8DR 16094666 Ki = 1.4 nM T24983 CP1VN8 16094667 EC50 = 8 nM T24983 C6IT7P 16094668 EC50 = 340 nM T24983 C9UKG0 16094670 EC50 = 70 nM T24983 C2XZ9B 16094671 EC50 = 240 nM T24983 CEBO78 16094672 EC50 = 145 nM T24983 C0ZV9M 16094674 EC50 = 36 nM T24983 CV30PU 16094675 EC50 = 1 nM T24983 C45TDZ 16094677 EC50 = 32 nM T24983 C1YJL4 16094678 EC50 = 160 nM T24983 CJ53QW 16094679 EC50 = 555 nM T24983 CG6IC9 16094680 EC50 = 95 nM T24983 CTF8D7 16094681 EC50 = 60 nM T24983 CD7NM6 16094682 EC50 = 134 nM T24983 C6LVM0 16094683 EC50 = 346 nM T24983 C80EYA 16094684 EC50 = 103 nM T24983 CH6TP1 16094685 EC50 = 294 nM T24983 CD6H5C 16094697 EC50 = 54 nM T24983 CGA63F 16094698 Ki = 1.3 nM T24983 CH36CE 16094699 EC50 = 9 nM T24983 CY38GV 16094700 EC50 = 8 nM T24983 C6FGX3 16094704 EC50 = 3.8 nM T24983 C45EKG 16094705 EC50 = 170 nM T24983 CT96PB 16094706 EC50 = 1290 nM T24983 CFU4K6 16094707 EC50 = 76 nM T24983 CDAL73 16094708 EC50 = 360 nM T24983 C8E6DX 16094709 EC50 = 473 nM T24983 CS1D0G 16121920 Ki = 6.4 nM T24983 CJ4E9C 16277250 Ki = 281 nM T24983 CZ2IS9 16660294 Ki > 10000 nM T24983 CRIH69 16744003 Ki = 225 nM T24983 C3D0FE 16744004 Ki = 426 nM T24983 CKDM79 16744005 Ki = 483 nM T24983 CQ1MG0 16744171 Ki = 507 nM T24983 CTI89R 16759249 Ki = 583 nM T24983 CF25CM 17449900 Ki = 0.28 nM T24983 CH7C6A 17461770 Ki = 3.981 nM T24983 C73MFP 17469721 Ki = 310 nM T24983 CPZJ30 17475863 Ki = 2.884 nM T24983 C7KP5T 17755866 Ki = 2258 nM T24983 CX7VE8 17755867 Ki = 60.15 nM T24983 CUW8S4 17755868 Ki = 422 nM T24983 C3KA6Z 17755875 Ki > 10000 nM T24983 C4N1LS 17755991 Ki = 4256 nM T24983 C6BE2Y 17755992 Ki > 10000 nM T24983 C10UQJ 17755999 Ki = 1103 nM T24983 C6WO9X 17756101 Ki = 271 nM T24983 CI9RW0 17756102 Ki = 2869 nM T24983 CDPT42 17756110 Ki > 10000 nM T24983 C0XG9B 17756212 Ki = 2763 nM T24983 C6JQ1K 17756213 Ki = 3751 nM T24983 CL5C3X 17888044 IC50 = 4 nM T24983 CZ78BE 17987129 Ki = 2700 nM T24983 C9PV8A 18180076 IC50 > 10000 nM T24983 C7Y9EN 18403576 Ki = 4.4 nM T24983 C9DQU7 18414156 Ki = 14.4 nM T24983 CO8U1V 18613655 IC50 = 7 nM T24983 CJ20BQ 18624462 Ki = 2.1 nM T24983 C6AOE8 19426635 IC50 = 302 nM T24983 CEN3L5 19964401 Ki = 6.2 nM T24983 C5IHG3 19964406 Ki = 140 nM T24983 C9VXS1 19964410 Ki = 5.6 nM T24983 CG8Z4W 20256387 Ki = 94 nM T24983 C8LD0M 20354789 Ki = 410 nM T24983 CP2R7D 21186098 IC50 = 8 nM T24983 CNR17B 21186102 IC50 = 57 nM T24983 CXY0P4 21186115 IC50 = 3 nM T24983 CY0QO4 21186124 IC50 = 6 nM T24983 C79MJX 21186138 IC50 = 7 nM T24983 CUJ4R9 21186143 IC50 = 17 nM T24983 CGY9F6 21186148 IC50 = 25 nM T24983 CRA23J 21186186 IC50 = 7 nM T24983 C18IWL 21186192 IC50 = 8 nM T24983 C5ER6Q 21186194 IC50 = 16 nM T24983 CLN86H 21219144 Ki = 27 nM T24983 C2M0HK 21219154 Ki = 15 nM T24983 C1GQY9 21219156 Ki = 18 nM T24983 C6LM2O 21219157 Ki = 0.39 nM T24983 C0W8PE 21219160 Ki = 32 nM T24983 CG4XF7 21219164 Ki = 3.1 nM T24983 C9S5XI 21219166 Ki = 40 nM T24983 CH83US 21219167 Ki = 17 nM T24983 C60TBU 21219173 Ki = 1200 nM T24983 CB3KF6 21219176 Ki = 1.2 nM T24983 C94BPG 21460314 Ki > 5000 nM T24983 C7MYT1 21462964 Ki = 1.8 nM T24983 C8GC6E 21462980 Ki = 7 nM T24983 C2D6ZX 21465540 Ki = 34 nM T24983 C3T5HF 21509921 Ki > 10000 nM T24983 CRE80D 21559988 Ki = 18000 nM T24983 CAH39X 21564536 Ki > 10000 nM T24983 CT7XG9 21830793 Ki = 21 nM T24983 CW90QB 21997225 Ki = 3.8 nM T24983 CLF09T 22065962 Ki = 56 nM T24983 COB35X 22065971 Ki = 1.9 nM T24983 CYCS06 22100932 Ki = 21 nM T24983 CM75DA 22100933 Ki = 26 nM T24983 CP48JW 22100940 Ki = 5 nM T24983 C68MQE 22100943 Ki = 8.1 nM T24983 CWH1R0 22100957 Ki = 8.4 nM T24983 C9TG8S 22100962 Ki = 44 nM T24983 CLCN93 22100964 Ki = 17 nM T24983 CC3LF7 22100965 Ki = 87 nM T24983 C90FER 22100968 Ki = 97 nM T24983 C9RUA4 22100970 Ki = 68 nM T24983 CVX19H 22727322 Ki = 774 nM T24983 CT45YC 22727323 Ki = 50 nM T24983 CL26HS 22727324 Ki = 33 nM T24983 CCS83F 22727331 Ki = 34 nM T24983 CS5J2U 22727332 Ki = 58 nM T24983 CAUK40 22727334 Ki = 541 nM T24983 CSCJ35 22727335 Ki = 198 nM T24983 CCIW17 22727346 Ki = 413 nM T24983 CS9IF2 22727347 Ki = 88 nM T24983 CFQ92N 22727351 Ki = 1697 nM T24983 CE2P3H 22727356 Ki = 346 nM T24983 C64UKQ 22727358 Ki = 117 nM T24983 CU6B2Z 22727361 Ki = 76 nM T24983 CAM3H4 22910005 Ki = 192 nM T24983 C04FIU 22953120 Ki = 206 nM T24983 CH5C7X 23288790 Ki = 1054 nM T24983 C0NI3J 23290944 Ki = 246 nM T24983 CLME84 23363843 Ki = 259 nM T24983 CEP65L 23364995 Ki = 9.3 nM T24983 CI4B6N 23642427 Ki = 250 nM T24983 C2BO0F 23928184 Ki > 3333 nM T24983 CDH38J 23992579 Ki = 52 nM T24983 C8TZY0 24810004 Ki = 640 nM T24983 CSCW01 24815434 Ki = 100 nM T24983 C0DYP7 24815883 Ki = 251.19 nM T24983 CN9AY0 24815976 Ki = 125.89 nM T24983 C2A0LT 24849462 Ki = 63.1 nM T24983 CKF9G6 24878061 EC50 = 230 nM T24983 C49GLI 24882561 Ki = 1.7 nM T24983 CAOF91 24894071 IC50 > 10000 nM T24983 C4IGH9 24936042 Ki = 13 nM T24983 CD0YW2 25070416 Ki = 29 nM T24983 C5QU0F 25070419 Ki = 33 nM T24983 CTN36E 25070740 Ki = 16 nM T24983 CGAZ01 25070742 Ki = 41 nM T24983 CKB23A 25071066 Ki = 130 nM T24983 CI8NL3 25071384 Ki = 57 nM T24983 C6F5SU 25071385 Ki = 7.1 nM T24983 CL7TN4 25071691 Ki = 5.3 nM T24983 C75ZIC 25071692 Ki = 5.7 nM T24983 C49ZFU 25072002 Ki = 1.3 nM T24983 CM28GQ 25072632 Ki = 4.4 nM T24983 C8OBV4 25072633 Ki = 0.69 nM T24983 CIT6G4 25072635 Ki = 18 nM T24983 CS1CI4 25072941 Ki = 4.3 nM T24983 C3CLH5 25072943 Ki = 16 nM T24983 C1XSD0 25072946 Ki = 78 nM T24983 CBKG34 25093832 Ki = 0.73 nM T24983 C2FY7C 25128757 Ki = 140 nM T24983 C5NW4M 25129807 Ki = 3007 nM T24983 CAV81B 25130157 Ki = 195 nM T24983 CFJ6Y9 25131876 Ki = 8.318 nM T24983 C67QCG 25132869 Ki = 364 nM T24983 CN61ZL 25139180 Ki = 3100 nM T24983 CLTF40 25139181 Ki = 4.3 nM T24983 CN32VX 25139329 Ki = 1100 nM T24983 C0LZ7B 25139335 Ki = 100 nM T24983 CW07GC 25139477 Ki = 69 nM T24983 CQD6N1 25139478 Ki = 1800 nM T24983 CN3S7R 25139479 Ki = 190 nM T24983 CSG25V 25139481 Ki = 670 nM T24983 CXDM41 25141533 Ki = 1230 nM T24983 CL84YJ 25141534 Ki = 2600 nM T24983 C4FXR9 25141535 Ki = 1920 nM T24983 CKBJ53 25141536 Ki > 10000 nM T24983 C8OGB1 25141538 Ki = 967 nM T24983 CX04LB 25142456 Ki = 90 nM T24983 COV83Z 25256814 Ki = 1.9 nM T24983 C7JZ2D 25256816 Ki = 1.3 nM T24983 CSW0O8 25895957 Ki = 3394 nM T24983 CPD3L4 25895959 Ki > 1000 nM T24983 C4MRQ0 27842480 IC50 > 50000 nM T24983 CE0PR6 30616772 Ki = 73 nM T24983 CAB4L3 30740059 Ki = 29 nM T24983 CM12QP 30743524 Ki = 726 nM T24983 CDY01I 30982708 Ki = 652 nM T24983 CY1O0S 41532205 Ki = 0.7 nM T24983 C2NS9O 42266974 Ki = 25.12 nM T24983 CG2KD8 42273483 Ki = 199.53 nM T24983 C0XMS9 42605994 Ki = 2000 nM T24983 CD61JW 42606339 Ki = 460 nM T24983 C0TN5O 42606573 Ki = 590 nM T24983 CQ37BN 42625290 Ki > 10000 nM T24983 CXB28J 42625293 Ki = 1290 nM T24983 CYM0J6 42625295 Ki = 1040 nM T24983 CD9RN1 42626103 Ki = 640 nM T24983 CTW8G4 42626171 Ki > 10000 nM T24983 C0P3JR 42626172 Ki = 2040 nM T24983 CZ19KX 42626240 Ki = 1900 nM T24983 CTL2I7 42626243 Ki > 5000 nM T24983 C98BKP 42626313 Ki = 2140 nM T24983 CRMZ20 42626317 Ki = 176 nM T24983 CRQ91B 42626318 Ki = 3430 nM T24983 CTYZ17 42626380 Ki = 455 nM T24983 C1JK6E 42626381 Ki = 1530 nM T24983 CEL6J0 44123782 Ki = 69 nM T24983 C6SG0O 44192200 Ki = 1418 nM T24983 CDO0I4 44214764 Ki = 17 nM T24983 CK01JN 44214765 Ki = 24 nM T24983 C9H3EV 44214766 Ki = 3 nM T24983 C7VWY4 44214767 Ki = 2 nM T24983 COS94W 44222483 Ki = 8.8 nM T24983 CNW3R8 44222488 Ki = 46 nM T24983 C1ST2I 44241718 Ki = 2.8 nM T24983 CJ8RW5 44249745 Ki = 170 nM T24983 C2FDB1 44250364 IC50 > 10000 nM T24983 C8MC0Q 44251387 IC50 > 10000 nM T24983 C5YEA8 44251388 IC50 > 10000 nM T24983 C0BSF6 44251389 IC50 > 10000 nM T24983 C1C0JQ 44263882 Ki = 1800 nM T24983 CQ13GA 44264622 Ki = 290 nM T24983 CMP0F2 44264623 Ki = 13 nM T24983 CHGO69 44264629 Ki = 140 nM T24983 CKD0E4 44264641 Ki = 7300 nM T24983 C41LTK 44264642 Ki = 3 nM T24983 CJI76B 44264644 Ki = 12.5 nM T24983 CS4YW5 44264682 Ki = 4 nM T24983 CCK6Z0 44264741 Ki = 23000 nM T24983 C6LNX8 44264742 Ki = 4500 nM T24983 CGA1W5 44269820 Ki = 92 nM T24983 C0C4QN 44269825 Ki = 260 nM T24983 C43LUM 44270444 Ki = 50 nM T24983 CWK09J 44270558 Ki = 2.692 nM T24983 C1WZB8 44273552 Ki = 1258.93 nM T24983 CU8Y6L 44273553 Ki = 125.89 nM T24983 C28FOS 44273715 Ki = 125.89 nM T24983 C2TN6O 44273720 Ki = 10 nM T24983 CQV2Y7 44273741 Ki = 19.95 nM T24983 CUK3H6 44273815 Ki = 316.23 nM T24983 C7Z6BK 44273855 Ki = 15.85 nM T24983 CT9ZA7 44273876 Ki = 158.49 nM T24983 CFBT63 44273877 Ki = 125.89 nM T24983 CPG2K5 44273882 Ki = 50.12 nM T24983 C7H4GN 44273884 Ki = 100 nM T24983 C5DAM2 44273887 Ki = 7.943 nM T24983 CDE2S1 44273896 Ki = 79.43 nM T24983 C2OMI3 44273897 Ki = 31.62 nM T24983 C3J0GV 44273908 Ki = 7.943 nM T24983 CY2G0T 44273912 Ki = 31.62 nM T24983 CG1L2J 44273920 Ki = 63.1 nM T24983 CMKG67 44273921 Ki = 63.1 nM T24983 CX5PF6 44273924 Ki = 12.59 nM T24983 CMW36L 44273925 Ki = 316.23 nM T24983 CUP96S 44273927 Ki = 12.59 nM T24983 CF46KT 44273928 Ki = 15.85 nM T24983 CE20CZ 44275807 Ki = 9772.37 nM T24983 CMI4G9 44275820 Ki = 683 nM T24983 CFP7Z8 44276050 Ki = 34 nM T24983 CE10KM 44276075 Ki = 21 nM T24983 CTM39J 44276079 Ki = 233 nM T24983 CQ8V6N 44276105 Ki = 465 nM T24983 C3AS0H 44276111 Ki = 51 nM T24983 CK32VR 44276155 Ki = 49 nM T24983 C9W5MA 44276170 Ki = 43 nM T24983 C84TMG 44278427 Ki = 11.6 nM T24983 CQ4N8P 44278456 Ki = 72 nM T24983 C4O6JE 44278458 Ki = 52 nM T24983 C2OG4D 44278479 Ki = 50 nM T24983 C2QOV4 44278496 Ki = 45 nM T24983 CXDF91 44278624 Ki = 45 nM T24983 CI37UT 44278788 Ki = 3.6 nM T24983 C3UK0D 44278789 Ki = 18 nM T24983 C9RJX8 44278829 Ki = 32 nM T24983 CX6ZN3 44278853 Ki = 74 nM T24983 C8Q5RI 44283757 Ki = 9.3 nM T24983 C1T2BY 44283889 Ki = 333 nM T24983 CZF8B5 44283891 Ki = 35.1 nM T24983 C5WHP1 44283941 Ki = 22.6 nM T24983 CCG7S8 44283963 Ki = 81.4 nM T24983 C2B0NQ 44284013 Ki = 8.6 nM T24983 CBSQ04 44300865 EC50 = 6.8 nM T24983 CQ5A2E 44301054 EC50 = 5.6 nM T24983 CZ59OL 44301157 Ki = 25.12 nM T24983 CNW2F3 44304314 IC50 = 4800 nM T24983 CCS0V1 44304600 IC50 = 290 nM T24983 CWJA31 44304603 Ki = 170 nM T24983 CK8QJ6 44304621 Ki = 170 nM T24983 CR9SB5 44304643 Ki = 650 nM T24983 CH6FM8 44304644 Ki = 1110 nM T24983 CGY80N 44304652 Ki = 390 nM T24983 CKBE16 44304814 Ki = 15500 nM T24983 C2C8LF 44307285 Ki > 1000 nM T24983 C7EJ1R 44307286 Ki > 1000 nM T24983 CJ2QR0 44307437 Ki > 1000 nM T24983 CFBL97 44307498 Ki > 1000 nM T24983 CTI68M 44307546 Ki > 1000 nM T24983 CFDV86 44307552 Ki = 59 nM T24983 CA3EG2 44307692 Ki > 1000 nM T24983 CP1QG5 44309688 Ki = 363 nM T24983 CKY68S 44309775 Ki = 1020 nM T24983 CU4V7O 44315403 Ki = 719 nM T24983 C6RF1P 44316315 Ki = 87 nM T24983 CV8WZ0 44318454 IC50 = 14.45 nM T24983 CXJL56 44318842 IC50 > 1000 nM T24983 CWUE26 44319102 Ki = 340 nM T24983 CV2UN7 44319361 Ki = 1200 nM T24983 CC2W9S 44319368 Ki = 390 nM T24983 CCD3V1 44319369 Ki = 440 nM T24983 CY9ZX7 44319370 Ki = 290 nM T24983 CG5E2U 44323763 Ki = 2.9 nM T24983 CY1I0M 44323780 Ki = 8.8 nM T24983 C5CP2K 44323851 Ki = 47 nM T24983 CVZ27T 44323870 Ki = 930 nM T24983 CHE75M 44323876 Ki = 2700 nM T24983 CAO54X 44323890 Ki = 300 nM T24983 C7Y5PV 44323894 Ki = 12 nM T24983 CW16JD 44324737 Ki > 1000 nM T24983 CA84SN 44324765 Ki > 1000 nM T24983 COA3H4 44324800 Ki > 1000 nM T24983 CY04JW 44324972 Ki > 1000 nM T24983 CCT67J 44324980 Ki = 7000 nM T24983 CCUZ21 44326212 Ki = 3.8 nM T24983 CV56DM 44326256 Ki = 55 nM T24983 C94UHT 44326285 Ki = 0.55 nM T24983 C2X9GN 44326324 Ki > 4067 nM T24983 C90PLN 44329483 IC50 > 10000 nM T24983 C5J3PW 44329749 Ki = 44.4 nM T24983 C5U1WN 44330292 Ki = 1293 nM T24983 C1WV6L 44330340 Ki = 2563 nM T24983 C4P1XE 44330386 Ki = 169 nM T24983 CDM14Y 44330387 Ki > 10000 nM T24983 CIWY10 44330417 Ki > 10000 nM T24983 CROD75 44330514 Ki = 138 nM T24983 C1UTG6 44330515 Ki = 1297 nM T24983 CFI52O 44330553 Ki = 11 nM T24983 C3UR9Q 44330554 Ki = 2866 nM T24983 C12EKB 44330564 Ki = 1563 nM T24983 COK95B 44330566 Ki = 168 nM T24983 C3DOY1 44330567 Ki = 14 nM T24983 CQRP49 44330574 Ki > 10000 nM T24983 CZPL05 44330585 Ki = 3548 nM T24983 C0RX1F 44330637 Ki = 507 nM T24983 C7CNK8 44330638 Ki = 462 nM T24983 C4JP8S 44330639 Ki = 4325 nM T24983 CJZQ05 44330640 Ki = 301 nM T24983 C98JGO 44330650 Ki = 425 nM T24983 CBL05A 44330692 Ki = 275 nM T24983 C26UAW 44330694 Ki = 97 nM T24983 C9JQK3 44332566 Ki = 27.2 nM T24983 C1E7KI 44332581 Ki = 297 nM T24983 CD7N6W 44332613 Ki > 400 nM T24983 C63TDB 44332686 Ki = 500 nM T24983 COG5D1 44332701 Ki = 137 nM T24983 C5XUT1 44335569 Ki = 290 nM T24983 C4QAZ1 44335635 Ki = 1600 nM T24983 CK1UB8 44335678 Ki = 40 nM T24983 CRD80K 44335721 Ki = 51 nM T24983 CIMQ72 44335722 Ki = 462 nM T24983 CO6YN8 44335739 Ki = 3 nM T24983 CRL68J 44335746 Ki = 12 nM T24983 C7AN0J 44335761 Ki = 25 nM T24983 CS4A3Z 44335795 Ki = 5 nM T24983 CL1BV7 44335796 Ki = 4 nM T24983 CJ98HN 44335798 Ki = 7 nM T24983 CT54MD 44335799 Ki = 6 nM T24983 C7FYS0 44335800 Ki = 15 nM T24983 C3I6KY 44335812 Ki = 2 nM T24983 C3YNI6 44335813 Ki = 29 nM T24983 C7Y2LT 44335816 Ki = 5 nM T24983 CB15TR 44335828 Ki = 12 nM T24983 CNZ0F5 44335829 Ki = 12 nM T24983 COS7V9 44335835 Ki = 5 nM T24983 CYIF05 44335847 Ki = 64 nM T24983 CM85JR 44335853 Ki = 11 nM T24983 C0A5DO 44335876 Ki = 8 nM T24983 CYE80K 44335877 Ki = 6 nM T24983 CLW0Z6 44335884 Ki = 6 nM T24983 C6WA4H 44335886 Ki = 7 nM T24983 CX8AZ4 44335889 Ki = 2 nM T24983 CCJ38R 44335893 Ki = 12 nM T24983 C0XR3S 44335896 Ki = 37 nM T24983 CQ2U5E 44335907 Ki = 15 nM T24983 C2D5HQ 44335908 Ki = 10 nM T24983 CR31UG 44335909 Ki = 11 nM T24983 C08FAK 44335918 Ki = 8 nM T24983 C85UNM 44335919 Ki = 3 nM T24983 CG6K4D 44335923 Ki = 6 nM T24983 C3EIN8 44335924 Ki = 7 nM T24983 C2A3OP 44335925 Ki = 5 nM T24983 CA2UE5 44335945 Ki > 1000 nM T24983 C5ILQ0 44335948 Ki = 5745 nM T24983 C6YM5Z 44335960 Ki = 6 nM T24983 CA1T9Z 44335971 Ki = 67 nM T24983 CT78OA 44335972 Ki = 134 nM T24983 C75EDP 44335973 Ki = 12 nM T24983 C5ZRM3 44335979 Ki = 771 nM T24983 C69XES 44335987 Ki = 50 nM T24983 CEV25H 44335991 Ki = 7 nM T24983 CSWA61 44335995 Ki = 4 nM T24983 CUK23N 44335996 Ki = 43 nM T24983 CZD10E 44335998 Ki = 522 nM T24983 CK1I5J 44336000 Ki = 4 nM T24983 C0AY1E 44336003 Ki = 726 nM T24983 COK93P 44336004 Ki = 81 nM T24983 C0QH8A 44336005 Ki = 37 nM T24983 C3QW4H 44336006 Ki = 3 nM T24983 CX2L3Z 44336012 Ki = 6.1 nM T24983 CR4SU0 44336027 Ki = 6 nM T24983 CG8U9R 44336030 Ki = 3 nM T24983 CSCX75 44336031 Ki = 7264 nM T24983 CHE0R6 44336035 Ki = 992 nM T24983 CQ38GM 44336036 Ki = 14 nM T24983 C3KV9L 44336045 Ki > 10000 nM T24983 C3EF1C 44336046 Ki = 1361 nM T24983 C5H1SL 44336047 Ki = 5 nM T24983 CRIF94 44336050 Ki = 4 nM T24983 CY60UT 44336051 Ki = 7 nM T24983 CL0HI9 44336052 Ki = 335 nM T24983 CO4M5K 44336055 Ki = 95 nM T24983 CJLR98 44336057 Ki = 1563 nM T24983 C4W8NC 44336059 Ki > 1000 nM T24983 C7OW8Y 44336061 Ki = 1.995 nM T24983 CYP35N 44336062 Ki = 139 nM T24983 CK1IQ0 44336074 Ki = 2 nM T24983 C6K9QY 44336075 Ki = 10 nM T24983 CD80AW 44336085 Ki = 59 nM T24983 CN4A2F 44336099 Ki = 7 nM T24983 CUQS13 44336100 Ki = 726 nM T24983 CP3HA8 44336105 Ki = 622 nM T24983 CK4H8R 44336108 Ki = 6 nM T24983 CDY2E4 44336109 Ki = 21 nM T24983 CFZ9U0 44336127 Ki = 549 nM T24983 CIB45H 44336138 Ki = 13 nM T24983 CJR1X5 44336154 Ki = 108 nM T24983 CX8EA2 44336172 Ki = 235 nM T24983 CJ4F0T 44336175 Ki = 6392 nM T24983 CJB61S 44336194 Ki = 235 nM T24983 CS7G8O 44336313 Ki = 27 nM T24983 C1YIQ4 44336314 Ki = 8 nM T24983 C26ZUF 44336352 Ki = 31 nM T24983 CFT4L1 44336552 Ki = 280 nM T24983 CS3TZ4 44336571 Ki = 230 nM T24983 CT3M2R 44337675 Ki > 4000 nM T24983 C2ECI8 44337709 Ki > 4000 nM T24983 C5S9WU 44337725 Ki = 541 nM T24983 C0ZH4Y 44338149 Ki = 868 nM T24983 CQ0ZF9 44338248 Ki = 172 nM T24983 C1I8XF 44339879 Ki = 25 nM T24983 C34CBZ 44339953 Ki = 7.4 nM T24983 CPF62D 44339984 Ki = 17 nM T24983 CIS79K 44339992 Ki = 2.7 nM T24983 C84OZX 44340084 Ki = 1.6 nM T24983 C9I7GN 44340097 Ki = 0.77 nM T24983 CBQ3D5 44340186 Ki = 200 nM T24983 CT5HC3 44340227 Ki = 1.2 nM T24983 C5HGU2 44340302 Ki = 500 nM T24983 CA71HQ 44340333 Ki = 2.5 nM T24983 CQPW26 44340376 Ki = 78 nM T24983 C3QW1F 44340415 Ki = 500 nM T24983 CD9ZS8 44342270 IC50 = 1690 nM T24983 C6N3XK 44345317 IC50 < 1000 nM T24983 CCU89V 44350664 Ki = 176.8 nM T24983 CZV3S0 44355355 Ki = 134 nM T24983 CNV5M9 44355433 Ki = 324 nM T24983 C9W5AB 44356064 Ki = 23 nM T24983 C9GB5E 44356253 Ki = 396 nM T24983 CJ80OW 44360984 Ki = 87 nM T24983 CS8K1A 44360992 Ki = 8.9 nM T24983 C3NZ7B 44361021 Ki = 67 nM T24983 CPO24U 44363755 IC50 = 120 nM T24983 C1VMY3 44364166 Ki = 5.8 nM T24983 C5JLD7 44369020 Ki = 3.95 nM T24983 C9ZB4M 44370009 Ki = 59 nM T24983 C81CTM 44370032 Ki = 30 nM T24983 C50OBQ 44370047 Ki = 11.7 nM T24983 C4JCY7 44370058 Ki = 26 nM T24983 C6PSR0 44371932 Ki = 2.6 nM T24983 CQ1IU6 44371980 Ki = 26 nM T24983 C2JFZ9 44371996 Ki = 180 nM T24983 CK6GM7 44371997 Ki = 1.5 nM T24983 CXZ6A7 44372009 Ki = 7.6 nM T24983 C4VLE2 44372153 Ki = 37 nM T24983 CJXL12 44372154 Ki = 87 nM T24983 C4O3LX 44372198 Ki = 29 nM T24983 CZV9O7 44372296 Ki = 19.5 nM T24983 C1SWI7 44372312 Ki = 110 nM T24983 CX2B6A 44372338 Ki = 2.8 nM T24983 CD5E1G 44374431 Ki = 1593 nM T24983 CK28HY 44374637 Ki = 121 nM T24983 C8EK9X 44374648 Ki = 621 nM T24983 CPL87U 44374827 Ki = 10 nM T24983 CEC54D 44374863 Ki = 12 nM T24983 CNF12S 44376209 Ki = 2 nM T24983 CG1H4I 44376230 Ki = 20 nM T24983 CGX1Z3 44376241 Ki = 18 nM T24983 C2UD1H 44376569 Ki = 1.7 nM T24983 CM57EJ 44376876 Ki = 1.6 nM T24983 C2S0TL 44376918 Ki = 1.7 nM T24983 CD2R5X 44376920 Ki = 316 nM T24983 CGX72S 44376921 Ki = 127 nM T24983 CYI39O 44380685 Ki = 140 nM T24983 CL1ER5 44380697 Ki = 180 nM T24983 C6B9PA 44380715 Ki = 19 nM T24983 CNSG64 44380716 Ki = 7000 nM T24983 C6MWD2 44380717 Ki = 250 nM T24983 CA5EW9 44380770 Ki = 200 nM T24983 C68MUE 44380774 Ki = 220 nM T24983 C4DGR5 44380785 Ki = 240 nM T24983 CUV90Q 44380802 Ki = 150 nM T24983 CCL54M 44380815 Ki = 47 nM T24983 CM01SN 44380816 Ki = 48 nM T24983 CT02DY 44380921 Ki = 990 nM T24983 C6PI1L 44381117 Ki = 340 nM T24983 CJ6I0B 44381118 Ki = 23 nM T24983 CBYQ74 44381146 Ki = 4200 nM T24983 C8GA2E 44381147 Ki = 130 nM T24983 C6SDO5 44381216 Ki = 1.5 nM T24983 C4OAD2 44381217 Ki = 1600 nM T24983 C67SRD 44381276 Ki = 3700 nM T24983 CKR9B8 44381279 Ki = 460 nM T24983 COB6T7 44381286 Ki = 3500 nM T24983 CZ7Q2X 44381424 Ki = 120 nM T24983 CQO5G1 44381432 Ki = 4400 nM T24983 CQ85AW 44389003 Ki > 5000 nM T24983 C8AG7U 44389016 Ki > 5000 nM T24983 CEO2W9 44393372 Ki = 42 nM T24983 CXP4Q7 44393393 Ki = 130 nM T24983 C6BZS0 44393403 Ki = 46 nM T24983 C86NED 44393411 Ki = 550 nM T24983 C9THO4 44393415 Ki = 31 nM T24983 CFKL54 44393594 Ki > 10000 nM T24983 C90ZPS 44393612 Ki > 10000 nM T24983 CMNR13 44393622 Ki > 10000 nM T24983 C1Q7UC 44393658 Ki = 174.5 nM T24983 CC6PB7 44393737 Ki = 113.5 nM T24983 C1EP9A 44393775 Ki = 14 nM T24983 CUZK03 44393797 EC50 = 96 nM T24983 CQAS90 44394590 Ki = 18 nM T24983 CTB7O0 44394599 Ki = 36 nM T24983 C4V1DZ 44394618 Ki = 8 nM T24983 C67SCU 44394629 Ki = 17 nM T24983 CGC24Z 44394636 Ki = 24 nM T24983 CSK9Z7 44394666 Ki = 2 nM T24983 CL8C1E 44394667 Ki = 3.4 nM T24983 CW0M6Y 44394675 Ki = 70 nM T24983 C1MC6J 44394742 Ki = 2 nM T24983 COD15M 44394743 Ki = 1.5 nM T24983 CBZU60 44394820 Ki = 17 nM T24983 COU0F6 44394884 Ki = 4 nM T24983 C8EC7R 44395709 Ki = 789 nM T24983 CF7I1C 44395711 Ki = 1015 nM T24983 C2KFE4 44395714 Ki = 345.3 nM T24983 C3RV6T 44395741 Ki = 7.6 nM T24983 C4B0OI 44397588 Ki = 1258.93 nM T24983 C5FP0R 44397589 Ki = 1584.89 nM T24983 CE3G8U 44397670 Ki = 794.33 nM T24983 C0E5HY 44400500 Ki = 3.3 nM T24983 CO8EU5 44400519 Ki = 0.6 nM T24983 CRX12E 44400553 Ki = 0.91 nM T24983 CIU18E 44400585 Ki = 0.37 nM T24983 CV8K2W 44400594 Ki = 21 nM T24983 C84RNU 44400626 Ki = 0.63 nM T24983 CY94SF 44400674 Ki = 0.52 nM T24983 C1B4QL 44403095 Ki > 10000 nM T24983 C1YL7Z 44403098 Ki > 10000 nM T24983 CFV98A 44403101 Ki > 10000 nM T24983 C6OY9S 44403102 Ki > 10000 nM T24983 CH4SX6 44403105 Ki > 10000 nM T24983 C12FIH 44403106 Ki > 10000 nM T24983 CQ4U2P 44403210 Ki = 34 nM T24983 CKE6T4 44403213 Ki = 44 nM T24983 CAJX39 44403214 Ki = 130 nM T24983 C61CNS 44403219 Ki = 100 nM T24983 C5AE9L 44403220 Ki = 76 nM T24983 CC6XM4 44403224 Ki = 97 nM T24983 C6JB4M 44403225 Ki = 9.9 nM T24983 CGE52H 44403232 Ki = 17 nM T24983 C4LKC1 44404394 Ki > 10000 nM T24983 C3EJ4G 44404396 Ki > 10000 nM T24983 CQU19N 44405414 Ki = 33 nM T24983 CJ3ED5 44405445 Ki = 52 nM T24983 CMB7E9 44405451 Ki = 22 nM T24983 CT5IP4 44405452 Ki = 15 nM T24983 C9YLW2 44405455 Ki = 14 nM T24983 C9Q7CS 44405466 Ki = 14 nM T24983 CCP9V7 44405469 Ki = 16 nM T24983 C68OGK 44405489 Ki = 14 nM T24983 CX7ER9 44405490 Ki = 21 nM T24983 C3I8EC 44405492 Ki = 4 nM T24983 CD29AT 44405522 Ki = 7 nM T24983 CYXC08 44405530 Ki = 78 nM T24983 CZ24HP 44408818 Ki = 43.4 nM T24983 CG87PW 44409290 Ki > 720 nM T24983 CR2CJ9 44412182 Ki = 1 nM T24983 CF9IW1 44412191 Ki = 5.248 nM T24983 C8FU9P 44412268 Ki = 9.9 nM T24983 C78RSG 44412269 Ki = 2.7 nM T24983 CKY57Q 44412458 Ki = 3.2 nM T24983 CK9FC8 44412468 Ki = 2.57 nM T24983 C63XKI 44412482 Ki = 0.4365 nM T24983 C2UBR0 44412494 Ki = 2.884 nM T24983 CMO83R 44414898 EC50 = 123 nM T24983 C4F1YB 44415054 EC50 = 18 nM T24983 CW35JZ 44415055 EC50 = 347 nM T24983 CU2FG6 44415569 Ki = 1810 nM T24983 CDU6Y5 44415593 Ki = 977 nM T24983 CH0BY5 44415672 Ki = 2000 nM T24983 CK59CO 44415689 Ki = 808 nM T24983 C7AZ5D 44415690 Ki = 1870 nM T24983 CEVY54 44415704 Ki = 4846 nM T24983 C89HPL 44417647 EC50 = 21 nM T24983 CVZ32C 44418745 EC50 = 111 nM T24983 CK17CY 44418747 EC50 = 60 nM T24983 C1EDC2 44418748 EC50 = 40 nM T24983 CCPO37 44419053 Ki = 30.9 nM T24983 CGL9E1 44419056 Ki = 151.36 nM T24983 CP5M3H 44419060 Ki = 57.54 nM T24983 CJ4EZ9 44419065 Ki = 0.5888 nM T24983 CIWX27 44419066 Ki = 3.236 nM T24983 C1TBA0 44426499 Ki = 71 nM T24983 CU38MT 44426509 Ki = 63 nM T24983 CYI94R 44426511 Ki = 167 nM T24983 CFB28T 44426512 Ki = 210 nM T24983 CS2GJ6 44426513 Ki = 222 nM T24983 C65ZXC 44427827 Ki = 4620 nM T24983 C9U8YT 44427831 Ki = 1490 nM T24983 COV6N3 44427842 Ki = 1460 nM T24983 CY0QJ2 44427970 Ki = 5048 nM T24983 C8XUP2 44431459 Ki = 329 nM T24983 COX39W 44431462 Ki = 116 nM T24983 CUA62V 44431463 Ki = 43 nM T24983 C67ATD 44431466 Ki = 44 nM T24983 CA5V1B 44431467 Ki = 119 nM T24983 C1D5PQ 44431468 Ki = 96 nM T24983 CR7XF9 44431471 Ki = 168 nM T24983 CP8LE6 44431472 Ki = 223 nM T24983 CJM5T8 44431473 Ki = 155 nM T24983 C9YX8U 44431474 Ki = 77 nM T24983 C45VTG 44431476 Ki = 69 nM T24983 CT2K7B 44431478 Ki = 54 nM T24983 CUQP47 44431479 Ki = 37 nM T24983 CRX04P 44431482 Ki = 103 nM T24983 C6CQ2A 44431483 Ki = 84 nM T24983 CIT48X 44431486 Ki = 16 nM T24983 C1D9LG 44431487 Ki = 31 nM T24983 CWZ62Y 44431488 Ki = 26 nM T24983 C04QWA 44431489 Ki = 11 nM T24983 CW07DT 44431490 Ki = 21 nM T24983 C2DV3O 44431492 Ki = 299 nM T24983 C7Z2RH 44431494 Ki = 326 nM T24983 C2B4WN 44436596 Ki = 8 nM T24983 CLV2E1 44436597 Ki = 22 nM T24983 C0LBO6 44436598 Ki = 0.45 nM T24983 CREV94 44436599 Ki = 12 nM T24983 CZ37MU 44436600 Ki = 110 nM T24983 CRW39P 44436601 Ki = 220 nM T24983 CG06FU 44436602 Ki = 16 nM T24983 C2GD0Z 44436603 Ki = 170 nM T24983 C1T9IF 44436605 Ki = 120 nM T24983 CBQ6F7 44436606 Ki = 330 nM T24983 C6ZJ1W 44436608 Ki = 40 nM T24983 C1OP6H 44436610 Ki = 190 nM T24983 CR6UK2 44436617 Ki = 35 nM T24983 CHTG80 44436618 Ki = 69 nM T24983 CI5K6A 44436621 Ki = 100 nM T24983 CG2X1D 44437896 Ki = 630 nM T24983 CX04CK 44437897 Ki = 1700 nM T24983 CC4V7G 44438186 Ki = 2820 nM T24983 CJ8W5C 44438197 Ki = 1550 nM T24983 CMGT04 44438199 Ki = 3540 nM T24983 C8C0HP 44438201 Ki = 1100 nM T24983 CJDT47 44438203 Ki = 3750 nM T24983 CU4AS8 44438204 Ki = 6090 nM T24983 CPAE72 44438206 Ki = 1360 nM T24983 CJM3K5 44438208 Ki = 679 nM T24983 CPH7V5 44438209 Ki = 1490 nM T24983 C6K3ZU 44438210 Ki = 129 nM T24983 CADG24 44438211 Ki = 3870 nM T24983 CLE5G1 44438213 Ki = 3930 nM T24983 C8ILG5 44438215 Ki = 2440 nM T24983 CFE50G 44438218 Ki = 2750 nM T24983 C3KS0B 44438219 Ki = 2293 nM T24983 CAQ5Y9 44438220 Ki = 348 nM T24983 C52KTZ 44438221 Ki = 365 nM T24983 C8LW2C 44438222 Ki = 2270 nM T24983 CF2WK6 44438223 Ki = 3930 nM T24983 CVT06Y 44438224 Ki = 3520 nM T24983 C4POI0 44438225 Ki > 20000 nM T24983 CO76KJ 44438226 Ki = 4450 nM T24983 CJZ69F 44438227 Ki = 1940 nM T24983 CS1H8X 44438228 Ki = 34.1 nM T24983 CEQ1L8 44438229 Ki = 1190 nM T24983 CUF21H 44438230 Ki = 2990 nM T24983 CU49FT 44438231 Ki = 677 nM T24983 CD89OH 44438232 Ki = 2146 nM T24983 C0VA9W 44438233 Ki = 167 nM T24983 CJSX04 44438234 Ki = 404 nM T24983 CWE9K4 44438235 Ki = 153 nM T24983 C5Q6PG 44438236 Ki = 5140 nM T24983 CWS8R5 44438237 Ki = 8890 nM T24983 C4BJ9F 44438238 Ki > 20000 nM T24983 CL4FV8 44438239 Ki = 319 nM T24983 CB1P9X 44454685 Ki = 82 nM T24983 CZJ8G6 44454707 Ki = 50 nM T24983 CC5SL3 44454709 Ki = 1.3 nM T24983 CD6M2F 44454710 Ki = 12 nM T24983 C5V3RI 44454711 Ki = 1.6 nM T24983 C1GKA2 44454734 Ki = 3.7 nM T24983 CBD62A 44454735 Ki = 1.8 nM T24983 CZL97F 44455426 Ki = 544 nM T24983 C12XGE 44456400 Ki = 5128.61 nM T24983 CL1F7V 44459452 Ki = 140 nM T24983 CF8DR7 44459463 Ki = 4.7 nM T24983 C9OY3U 44517726 Ki = 158.49 nM T24983 CT85QK 44538690 Ki = 320 nM T24983 C16HEZ 44555445 Ki > 10000 nM T24983 C5SP0Z 44578445 Ki = 2100 nM T24983 CVR7A5 44578446 Ki = 520 nM T24983 CRCH48 44582675 Ki = 442 nM T24983 CEJ4R8 44582676 Ki = 174 nM T24983 C5QB4K 44582678 Ki = 2708 nM T24983 C01RCI 44582705 Ki = 923 nM T24983 C8S1HM 44591042 Ki = 277.5 nM T24983 CTQ1D6 44591043 Ki = 816.5 nM T24983 C5C6GE 44591045 Ki = 18.6 nM T24983 C4YRD3 44591086 Ki = 7873 nM T24983 CS5Q7A 44591087 Ki = 583.7 nM T24983 CPA4R6 44591088 Ki = 513 nM T24983 CF20PY 44591089 Ki = 1213 nM T24983 C1SN7Y 44593709 Ki = 52 nM T24983 C0DLU3 45109862 IC50 = 1845 nM T24983 CPR46X 45265656 Ki = 176.8 nM T24983 CM2YT9 45267409 Ki = 39 nM T24983 CCLR12 45267435 Ki = 6.4 nM T24983 C71SGH 45268292 Ki = 3.4 nM T24983 CL0CW7 45268293 Ki = 25 nM T24983 C0F9UT 45269161 Ki = 120 nM T24983 CQP0N3 45269168 Ki = 16 nM T24983 CJ18ZC 45270021 Ki = 70 nM T24983 CL42RS 45270813 Ki = 960 nM T24983 C5RX4W 45270861 Ki = 360 nM T24983 C4AJP5 45271653 Ki = 12 nM T24983 C13RSZ 45271691 Ki = 66 nM T24983 CZ8VO5 45272537 Ki = 14 nM T24983 CGZW61 45272580 Ki = 66 nM T24983 C9M6XP 45273045 Ki = 1.2 nM T24983 C19BMF 45273442 Ki = 21 nM T24983 C7VR4A 45273443 Ki = 3.8 nM T24983 CZ71RN 45278805 IC50 = 984 nM T24983 CZN6M7 45278882 IC50 = 645 nM T24983 CKQG15 45361874 Ki = 2.23 nM T24983 CYJ7P8 45379368 Ki > 10000 nM T24983 CU2CA7 45379369 Ki = 39.1 nM T24983 CT3K8Y 45379370 Ki = 225 nM T24983 CT3A1Q 45379373 Ki > 10000 nM T24983 C8TRE1 45379377 Ki > 10000 nM T24983 CML67J 45379515 Ki > 10000 nM T24983 C0SF6L 45482151 Ki = 47 nM T24983 CXC65S 45482152 Ki = 5.7 nM T24983 C8TE2Y 45482153 Ki = 240 nM T24983 C9LX5P 45482169 Ki = 28 nM T24983 CJD2A3 45482180 Ki = 1800 nM T24983 C0CHF4 45482789 IC50 = 2650 nM T24983 CO1M6P 45483654 Ki = 3400 nM T24983 CIV3Q4 45483655 Ki = 850 nM T24983 CLBT94 46190877 Ki = 630.96 nM T24983 CSV1P2 46216855 Ki = 10000 nM T24983 C68EGY 46225320 Ki = 630.96 nM T24983 CGH0M1 46225334 Ki = 251.19 nM T24983 COFU37 46225335 Ki = 398.11 nM T24983 C9XTG3 46225336 Ki = 794.33 nM T24983 C96LBQ 46225337 Ki = 1000 nM T24983 CS6Y9W 46225581 Ki = 251.19 nM T24983 C78DON 46225582 Ki = 7.943 nM T24983 CC8E3T 46225583 Ki = 199.53 nM T24983 CML42B 46225584 Ki = 2511.89 nM T24983 CY7NM6 46227242 Ki > 10000 nM T24983 CR9S7B 46227243 Ki > 10000 nM T24983 C9A8FV 46227273 Ki = 6644 nM T24983 CL3KU2 46227284 Ki > 10000 nM T24983 CS4O6A 46227317 Ki = 2565 nM T24983 CE1L6H 46227320 Ki > 10000 nM T24983 CSQ9D5 46227325 Ki > 10000 nM T24983 CDI10H 46231541 Ki > 10000 nM T24983 C9KI4E 46231646 Ki > 10000 nM T24983 C8SFI5 46231768 Ki > 10000 nM T24983 C1EW4S 46231782 Ki = 4830 nM T24983 C6JM5T 46231784 Ki = 3987 nM T24983 CD6IC3 46231845 Ki = 10000 nM T24983 C38WBY 46231846 Ki = 5972 nM T24983 C0A7GW 46231847 Ki = 6281 nM T24983 CVT82S 46231848 Ki = 10000 nM T24983 C9W1US 46231924 Ki = 7506 nM T24983 CL7WX9 46231925 Ki = 5886 nM T24983 CVG26Z 46231926 Ki = 8344 nM T24983 CKJ09A 46231927 Ki = 10000 nM T24983 C2BX8U 46231994 Ki = 10000 nM T24983 C7FD2G 46231995 Ki = 10000 nM T24983 CYV52A 46232066 Ki = 10000 nM T24983 C5TC2S 46830335 IC50 > 10000 nM T24983 C1K7FL 46830336 IC50 > 10000 nM T24983 C1N4KX 46842383 IC50 > 10000 nM T24983 CC62SX 46866711 IC50 > 10000 nM T24983 C03LTM 46869265 Ki = 2650000 nM T24983 CB8GE1 46884818 IC50 > 10000 nM T24983 C4MQ0A 46884856 IC50 > 10000 nM T24983 CCNT25 46884898 IC50 > 10000 nM T24983 C3MSG2 46885027 IC50 > 10000 nM T24983 CB7XI0 46885213 IC50 = 3800 nM T24983 CRW2I9 46893146 Ki = 2.3 nM T24983 CV9E5Y 46912547 Ki = 60.4 nM T24983 C34ILU 46912548 Ki = 129 nM T24983 CGSN70 46917563 Ki = 42 nM T24983 CEH10Y 46917637 Ki = 22 nM T24983 CUTX67 46934428 IC50 > 1000 nM T24983 CESC01 49782398 Ki = 0.72 nM T24983 C8BWU1 49782600 Ki = 20 nM T24983 C6I0NJ 49782601 Ki = 39 nM T24983 C20CVH 49782602 Ki = 30 nM T24983 CY4FW1 49782603 Ki = 61 nM T24983 CXJ59F 49782604 Ki = 30 nM T24983 CD9ZH7 49782836 Ki = 120 nM T24983 CL1J4C 49782837 Ki = 120 nM T24983 CB53QP 49782841 Ki = 880 nM T24983 CENR09 49783039 Ki = 300 nM T24983 CZ5G9J 49783040 Ki = 23 nM T24983 C98JVY 49783041 Ki = 170 nM T24983 CRML65 49783042 Ki = 220 nM T24983 COM8D5 49798797 Ki = 634 nM T24983 C9ZYH8 49798799 Ki = 937 nM T24983 C4TXW8 49798812 Ki = 245 nM T24983 C9KOV8 49798833 Ki = 377 nM T24983 C6LP9T 49798835 Ki = 94.5 nM T24983 C6RE1F 49798837 Ki = 40.4 nM T24983 CMQ23B 49798839 Ki = 163 nM T24983 C2WZ9Y 49798853 Ki = 72.6 nM T24983 CU34RI 49798855 Ki = 492 nM T24983 CM86YK 49798857 Ki = 945 nM T24983 CTDN46 49798874 Ki = 978 nM T24983 CO4K6F 49798877 Ki > 2000 nM T24983 C69EKV 49798878 Ki > 3500 nM T24983 CWQ9Y1 49798879 Ki = 700 nM T24983 CV1S3H 49799687 Ki = 53.4 nM T24983 CBR67S 49799691 Ki > 10000 nM T24983 C5A6TG 49799693 Ki = 344 nM T24983 CZ8A2G 49799695 Ki = 1390 nM T24983 CCV35T 49799709 Ki = 668 nM T24983 CLY02B 49799713 Ki = 2230 nM T24983 CDTS15 49799715 Ki = 620 nM T24983 C6IW4Q 49862238 Ki = 148 nM T24983 C9KIU1 49864289 IC50 > 10000 nM T24983 CHO9C0 49864292 IC50 > 10000 nM T24983 C90MTG 49864602 IC50 > 10000 nM T24983 C5BCS4 49864722 IC50 > 10000 nM T24983 CKZO79 49864723 IC50 > 10000 nM T24983 C74LZS 49864724 IC50 > 10000 nM T24983 C2RY0J 50878551 Ki > 10000 nM T24983 C1W6TV 50898777 Ki > 10000 nM T24983 CXMZ73 50898778 Ki > 10000 nM T24983 C8TA1J 51003550 IC50 > 10000 nM T24983 CQ1UJ7 51003551 IC50 = 5522 nM T24983 CGMI37 51003586 IC50 > 10000 nM T24983 CE4KP1 51050257 Ki > 10000 nM T24983 CU3C4O 51353676 Ki = 890 nM T24983 C1LHZ4 51353678 Ki = 990 nM T24983 CWFU41 51353989 Ki = 246 nM T24983 CW8LE6 51353992 Ki = 890 nM T24983 C2DG1Z 51354275 Ki = 182 nM T24983 CT8MC6 51354277 Ki = 1400 nM T24983 COD5H3 51354851 Ki = 2100 nM T24983 C42GMN 52937680 Ki = 230 nM T24983 C96LHK 52937776 Ki = 59 nM T24983 C30RKG 52937777 Ki = 190 nM T24983 C78FZD 52937871 Ki = 6300 nM T24983 CS5I2W 52940985 Ki = 10 nM T24983 C4PQ7Z 52942934 IC50 = 9 nM T24983 C09RJS 52943802 Ki = 45 nM T24983 CT51OC 52945819 Ki = 17 nM T24983 C19ZKQ 52946556 Ki = 11.3 nM T24983 CUV0G4 52947756 Ki = 19 nM T24983 C03JEZ 53248159 Ki = 3090 nM T24983 C2UKM3 53248209 Ki = 5340 nM T24983 CVD7E5 53248212 Ki = 1490 nM T24983 CX6KG9 53248213 Ki = 3360 nM T24983 C63MQD 53248256 Ki = 3180 nM T24983 CGY45S 53248361 Ki = 329 nM T24983 CE9L8G 53248365 Ki = 890 nM T24983 CC78FG 53248673 Ki = 185 nM T24983 CL3WJ1 53248675 Ki = 30.1 nM T24983 CG6T2N 53248677 Ki = 31.9 nM T24983 C61DNP 53320009 IC50 = 3613 nM T24983 C9ZDR5 53320010 IC50 = 1789 nM T24983 CQLK01 53322638 IC50 > 10000 nM T24983 C32YWL 53324045 Ki = 58 nM T24983 CRQF15 53325242 Ki = 385 nM T24983 C0UC1W 53326601 Ki = 896 nM T24983 CS5Z7X 53327908 Ki = 3.4 nM T24983 CLZ09P 53359025 Ki = 93 nM T24983 CPQ1E2 53361301 Ki = 15 nM T24983 CABK98 53361302 Ki = 7.2 nM T24983 CK0M7F 53363109 Ki = 3.3 nM T24983 CG24FV 53363110 Ki = 13 nM T24983 C28MPE 53363199 Ki = 8.4 nM T24983 CN3C4E 53363200 Ki = 6.4 nM T24983 CYW7M4 53363201 Ki = 12 nM T24983 C6EU7I 53363202 Ki = 19 nM T24983 CMI25H 53364083 Ki = 14 nM T24983 C1UWI5 53364153 Ki = 5.4 nM T24983 C78PUJ 53364154 Ki = 19 nM T24983 CRB76A 53364155 Ki = 11 nM T24983 CZV06L 53364225 Ki = 6.8 nM T24983 CQ7PX0 53364226 Ki = 12 nM T24983 CCA02T 53364227 Ki = 19 nM T24983 CMOZ61 53475319 Ki = 45 nM T24983 CKND43 54580905 Ki = 3.4 nM T24983 CF6G4L 54580906 Ki = 3.3 nM T24983 CHNI24 54581963 Ki = 3 nM T24983 CM5TK0 54581964 Ki = 2.9 nM T24983 C8AT1S 54583897 Ki = 2.8 nM T24983 CW9Z2J 54583898 Ki = 4.1 nM T24983 CL23NI 54585810 Ki = 9.8 nM T24983 CW1I5B 54585811 Ki = 6.1 nM T24983 CQ3AR0 56589560 Ki = 64.1 nM T24983 C4XGR3 56589561 Ki = 4861 nM T24983 C9PHZ3 56594402 Ki > 10000 nM T24983 C82IVX 56594533 Ki > 10000 nM T24983 CT4J5C 56594534 Ki = 408 nM T24983 C6W1RA 56649648 Ki = 71 nM T24983 C2SW7J 56649649 Ki = 84 nM T24983 CQTR49 56649650 Ki = 92 nM T24983 CJ57IF 56658006 Ki = 1352 nM T24983 CTWV58 56658008 Ki = 201 nM T24983 C1CJ8P 56664948 Ki = 1029 nM T24983 C26RNX 56664950 Ki = 286 nM T24983 CRPA72 56664952 Ki = 234 nM T24983 CW7F5G 56675269 Ki = 359 nM T24983 CC2B8F 56678599 Ki = 1311 nM T24983 C28ECA 56681925 Ki = 865 nM T24983 CLX25U 56681927 Ki = 27.2 nM T24983 CFE60O 56833378 Ki = 34 nM T24983 C04VKH 56833379 Ki = 660 nM T24983 CAS80D 56833463 Ki = 84 nM T24983 CUXP15 56833464 Ki = 40 nM T24983 C6DEW7 56837419 Ki = 78 nM T24983 CZ1WY0 56837634 Ki = 130 nM T24983 CKJ2U0 56837635 Ki = 140 nM T24983 CZP6E4 56837636 Ki = 38 nM T24983 CXJ7R9 56926585 Ki = 4.2 nM T24983 CH1S9B 56926586 Ki = 7.3 nM T24983 CJ42HS 56926587 Ki = 15 nM T24983 CB0P9N 56944383 Ki = 14 nM T24983 C1TC7Q 56963799 Ki > 10000 nM T24983 CQ5TP0 56964794 Ki = 42 nM T24983 CDGZ96 57326583 Ki = 210 nM T24983 C20ILW 57326584 Ki = 798 nM T24983 C0QM2U 57390115 Ki = 220 nM T24983 CZ12PI 57390116 Ki = 48 nM T24983 CRG2X7 57390117 Ki = 240 nM T24983 CR9L2W 57390118 Ki = 68 nM T24983 C26DAH 57390119 Ki = 190 nM T24983 C0T9UH 57391895 Ki = 82 nM T24983 CPN87T 57391896 Ki = 160 nM T24983 C64AWK 57391897 Ki = 70 nM T24983 C1M4PZ 57393627 Ki = 360 nM T24983 C7E4BW 57393628 Ki = 77 nM T24983 CGWK23 57393634 Ki = 5400 nM T24983 C39YHG 57395340 Ki = 250 nM T24983 C35RST 57395341 Ki = 45 nM T24983 C5YZM2 57398875 Ki = 140 nM T24983 CI9XS8 57400556 Ki = 64 nM T24983 C20IPH 57400557 Ki = 160 nM T24983 CU0C3D 57400562 Ki = 2400 nM T24983 CO04CI 57402365 Ki = 140 nM T24983 C27OEI 57402366 Ki = 100 nM T24983 CFJ27E 57402787 Ki = 51 nM T24983 CH3T2M 57587922 Ki = 292 nM T24983 C4MV2N 60149678 Ki = 70 nM T24983 CRH49P 60167309 Ki = 140 nM T24983 COHK72 60167451 Ki = 1698.24 nM T24983 C30SVG 60167452 Ki = 162 nM T24983 CKM14W 69432471 Ki = 60 nM T24983 C34GMW 69599704 Ki > 10000 nM T24983 CC43QK 71151588 Ki = 7.1 nM T24983 C0O5KW 71449034 Ki = 510 nM T24983 C4K5YQ 71449110 Ki = 23.9 nM T24983 CG06AP 71449737 Ki = 15 nM T24983 CE6YD5 71450707 Ki = 3.8 nM T24983 CBP03H 71450812 Ki = 20 nM T24983 C67MOE 71450871 Ki = 32 nM T24983 CDI84E 71450922 IC50 > 10000 nM T24983 CK8HN7 71452737 EC50 = 594 nM T24983 C7SQ0I 71453386 Ki = 252 nM T24983 C4X9KY 71454294 Ki = 4.6 nM T24983 CA65OQ 71454295 Ki = 0.79 nM T24983 C8YKT4 71454405 Ki = 150 nM T24983 CFWR57 71454487 Ki > 800 nM T24983 CQSA61 71455082 Ki = 550 nM T24983 C8YH0J 71455083 Ki = 55 nM T24983 CD4HQ6 71456045 Ki = 0.71 nM T24983 CD78KL 71456046 Ki = 1.5 nM T24983 CM30AR 71456214 Ki = 150 nM T24983 CZ7XH9 71456235 Ki = 890 nM T24983 C1H3MD 71456253 EC50 = 601 nM T24983 C82HSE 71456889 Ki = 69 nM T24983 C1PHO6 71456890 Ki = 807 nM T24983 CSX5J0 71457844 Ki = 1.9 nM T24983 CNM83V 71457956 Ki = 150 nM T24983 CNQ5B6 71458040 Ki = 6.5 nM T24983 C84QJC 71458071 Ki = 18 nM T24983 CI6H3T 71458739 Ki = 184 nM T24983 CI6OW4 71459759 Ki = 16 nM T24983 CSY3U1 71459760 Ki = 19 nM T24983 CD10CQ 71459761 Ki = 6 nM T24983 CG0WO9 71459954 Ki > 5000 nM T24983 CMOF94 71460561 Ki = 35 nM T24983 C9ESJ4 71461481 Ki = 9.5 nM T24983 CHJ27Z 71462265 Ki = 56.8 nM T24983 CLP8D6 71462266 Ki = 291 nM T24983 CKX5O8 71463061 Ki > 10000 nM T24983 C82GIQ 71463207 Ki = 2.4 nM T24983 CO3E4N 71583848 Ki = 2.5 nM T24983 C8N2ML 71583849 Ki = 45 nM T24983 CJ8FA6 71652196 Ki = 34 nM T24983 C5VH2Z 71657942 Ki = 608 nM T24983 CY9ES0 71657943 Ki = 372 nM T24983 CU41CZ 71657944 Ki = 429 nM T24983 C0S6YV 71657945 Ki = 522 nM T24983 CX52VK 71657946 Ki = 728 nM T24983 C6KJW5 71657947 Ki = 350 nM T24983 C6AQG0 71658072 Ki = 159 nM T24983 CQ3W7X 71658073 Ki = 188 nM T24983 CE3V4J 71658074 Ki = 161 nM T24983 C40XRK 71658075 Ki = 297 nM T24983 CPI8E9 71658076 Ki = 342 nM T24983 CC1U6V 71658077 Ki = 748 nM T24983 C8LX4D 71658203 Ki = 657 nM T24983 CVX3G1 71658204 Ki = 177 nM T24983 C29STX 71658205 Ki = 403 nM T24983 CR0EN8 71658206 Ki = 641 nM T24983 CF41PZ 71658207 Ki = 830 nM T24983 C7LMV3 71658208 Ki = 441 nM T24983 CIAR53 71658338 Ki = 706 nM T24983 CZ65JA 71659909 Ki = 187 nM T24983 C65JRT 71717830 Ki = 1200 nM T24983 CQO30I 71733932 Ki = 5.8 nM T24983 C93QMB 71733935 Ki = 11 nM T24983 COM72V 71734028 Ki = 37 nM T24983 C4S5WD 71734029 Ki = 14 nM T24983 C2ZX1W 71734031 Ki = 5.3 nM T24983 C7GDW5 71734126 Ki = 110 nM T24983 CQJ8P4 71734127 Ki = 22 nM T24983 CR53GT 71734129 Ki = 4.8 nM T24983 C31THM 72164180 Ki = 49.9 nM T24983 C56VLM 72164181 Ki = 7.4 nM T24983 CD8A9K 72164182 Ki = 78 nM T24983 C4C0BH 72164183 Ki = 152 nM T24983 CQU81Y 72164299 Ki = 4.4 nM T24983 CF0H7K 72164300 Ki = 31 nM T24983 C7WM5U 72164301 Ki = 11 nM T24983 C4HO2U 72164302 Ki = 6.2 nM T24983 CMPS48 72190766 Ki = 480 nM T24983 C4E8TR 72191064 Ki = 386.7 nM T24983 C85FKU 72191065 Ki = 394.8 nM T24983 CNPA07 72191066 Ki = 532.5 nM T24983 CQL1T2 72191067 Ki = 1898.2 nM T24983 CI2M7H 72191068 Ki = 426.4 nM T24983 C7AOY4 72198754 IC50 = 65 nM T24983 C4M7KP 72198756 IC50 > 100 nM T24983 C3TOA8 72205043 Ki = 100 nM T24983 CO53SR 72205044 Ki = 1500 nM T24983 C5UN3D 72205045 Ki = 330 nM T24983 CU4W5M 72205046 Ki = 800 nM T24983 CZP67J 72205222 Ki = 1180 nM T24983 C0U5RS 72544566 Ki = 20 nM T24983 CVY4I0 72544787 Ki = 32 nM T24983 C8UM5H 72544789 Ki = 23 nM T24983 CVU61Z 72545007 Ki = 150 nM T24983 CR6HY3 72545008 Ki = 680 nM T24983 CC25RP 72545009 Ki = 500 nM T24983 CW9OZ7 72545010 Ki = 340 nM T24983 C14DJV 72545011 Ki = 14 nM T24983 C4E5ZF 72545238 Ki = 5.1 nM T24983 CY7J8U 72545239 Ki = 100 nM T24983 CU72QA 72545240 Ki = 16 nM T24983 C3IM9Y 72737725 Ki = 1070 nM T24983 CC01EJ 72737728 Ki = 46 nM T24983 C6XYJ3 72737730 Ki = 65 nM T24983 CI9K6Y 72737734 Ki = 110 nM T24983 C6IF9H 72737744 Ki = 43 nM T24983 C0PI2G 72737750 Ki = 320 nM T24983 CY9U0X 72737767 Ki = 81 nM T24983 C5CX2V 72737772 Ki = 1020 nM T24983 CC65OA 73213195 Ki > 10000 nM T24983 CW83DK 73213196 Ki = 1230.27 nM T24983 CCV91B 73346042 Ki = 71 nM T24983 CK0HR9 73346334 Ki > 10000 nM T24983 C5QYH1 73347474 Ki = 30 nM T24983 CY60RD 73347826 Ki > 10000 nM T24983 CPN5T8 73350334 IC50 = 110 nM T24983 C9NAE5 73350335 IC50 = 70 nM T24983 C8RM2F 73350336 IC50 = 850 nM T24983 C10BUE 73353325 IC50 = 470 nM T24983 CCIT57 73353534 Ki = 59 nM T24983 C7IA8U 73354844 IC50 = 740 nM T24983 CX4Q3F 73354845 IC50 = 30 nM T24983 CO1VP6 73356382 IC50 = 30 nM T24983 C2E7QW 75201901 Ki = 4500 nM T24983 C8IDL3 75306277 Ki = 199.53 nM T24983 CTH23U 76309672 Ki = 47 nM T24983 C08KCY 76309673 Ki = 2.9 nM T24983 C5OYN0 76311261 Ki = 284 nM T24983 C2VAS4 76311270 Ki = 565 nM T24983 CZFW19 76314267 Ki = 14.3 nM T24983 CIYJ90 76316875 Ki = 1.7 nM T24983 CQM65S 76318472 Ki = 360 nM T24983 CGZP35 76318476 Ki = 444 nM T24983 CD16XI 76320592 Ki = 2.6 nM T24983 CIB40D 76321554 Ki = 1.549 nM T24983 CS9F1X 76321556 Ki = 9.55 nM T24983 C97LOB 76325150 Ki = 0.955 nM T24983 CCR29U 76325152 Ki = 31.62 nM T24983 CLP59V 76325156 Ki = 5.012 nM T24983 C3K6UP 76325763 Ki = 162 nM T24983 C17YTI 76328715 Ki = 22.91 nM T24983 CHRD95 76331467 Ki = 14.7 nM T24983 CSW58A 76336021 Ki = 47.86 nM T24983 C1UZ5J 76441180 Ki = 200 nM T24983 C8EWX5 85658088 Ki = 1174 nM T24983 CT8HK6 90389439 Ki = 6300 nM T24983 CU9ED1 90389592 Ki = 3820 nM T24983 CLFV10 90644226 Ki = 47 nM T24983 CZ7LD8 90644227 Ki = 35 nM T24983 C35GPQ 90644228 Ki = 89 nM T24983 CZI30L 90644230 Ki = 9.3 nM T24983 CUO0J6 90644928 Ki > 9000 nM T24983 CF9HI4 90644929 Ki > 14000 nM T24983 CX2WE7 90644930 Ki > 3000 nM T24983 C4MUI2 90664601 IC50 > 10000 nM T24983 CHT7D5 90664962 IC50 = 3942 nM T24983 CCV0I4 92640710 Ki > 100000 nM T24983 C92NBD 92984956 Ki = 110 nM T24983 C7PNG8 92988697 Ki = 10.4 nM T24983 C9NR7H 93601125 Ki = 43 nM T24983 COA3U6 102262219 Ki = 3300 nM T24983 CE6Z3M 109030343 Ki = 32.2 nM T24983 CC1P6O 109030515 Ki = 33 nM T24983 C2I0HB 118643968 Ki = 1750 nM T24983 CJS6B2 118709159 Ki = 24 nM T24983 C9XDM6 118709160 Ki = 33 nM T24983 CQ9C5S 118709161 Ki = 41 nM T24983 C1YRW4 118709162 Ki = 360 nM T24983 CPL69Z 118709163 Ki = 300 nM T24983 CGAB49 118709164 Ki = 520 nM T24983 C3SX4Z 118709165 Ki = 490 nM T24983 CC7FW6 118709166 Ki = 2200 nM T24983 CRMK67 118709167 Ki = 490 nM T24983 CW4YS6 118709168 Ki = 1400 nM T24983 CY3BR2 118709169 Ki = 570 nM T24983 CIX72C 118709170 Ki = 160 nM T24983 C2O8BG 118709171 Ki = 850 nM T24983 COV8K7 118709172 Ki = 130 nM T24983 CJZD82 118709173 Ki = 33 nM T24983 C16WQU 118709174 Ki = 29 nM T24983 C4E5MK 118709175 Ki = 8.7 nM T24983 CFV2M0 118709176 Ki = 19 nM T24983 C08TAX 118709177 Ki = 89 nM T24983 CYNM75 118709178 Ki = 41 nM T24983 CJZ7G0 118709179 Ki = 46 nM T24983 CE89TI 118714552 Ki = 28 nM T24983 C8M1VO 118719792 Ki = 486 nM T24983 CG0O3Q 118719795 Ki = 875 nM T24983 CUHT71 118719796 Ki = 186 nM T24983 CR0FM7 118719797 Ki = 90 nM T24983 CPX2Y1 118719798 Ki = 395 nM T24983 C0KH8S 118719799 Ki = 163 nM T24983 CWO13F 118719807 Ki = 758 nM T24983 CUH0A6 118719810 Ki = 227 nM T24983 CT8KO4 118719925 Ki = 74.13 nM T24983 C16DHZ 118719926 Ki = 4.365 nM T24983 CLA06I 118719927 Ki = 100 nM T24983 C1PKR0 121304441 Ki = 5888.44 nM T24983 CW68KD 121304458 Ki > 100000 nM T24983 C35WTP 122177641 Ki = 30 nM T24983 C8OS7B 122177642 Ki = 180 nM T24983 CV2AT4 122177644 Ki = 290 nM T24983 CB16GY 122177645 Ki = 9.4 nM T24983 CP6VX4 122180568 Ki = 299 nM T24983 CU0L3S 122180569 Ki = 329 nM T24983 C87MAH 122180570 Ki = 353 nM T24983 CY9BN0 122180571 Ki > 1000 nM T24983 CS9NY8 122180572 Ki > 2000 nM T24983 CAL57I 122180573 Ki = 4450 nM T24983 CZ72GE 122180574 Ki = 510 nM T24983 CZ4M2F 122180575 Ki = 232 nM T24983 C03CGT 122180576 Ki = 588 nM T24983 C2X3ZW 122180610 Ki = 222 nM T24983 CRMS80 122180611 Ki = 269 nM T24983 CWO2Y4 122180612 Ki = 425 nM T24983 C2DZ0K 122180613 Ki > 1000 nM T24983 CH81IV 122180614 Ki > 20000 nM T24983 C1EPB8 122180615 Ki > 2000 nM T24983 CV26IM 122180616 Ki > 1000 nM T24983 CQ0L6Z 122180617 Ki > 10000 nM T24983 CVX5Y3 122180618 Ki > 2000 nM T24983 CEGV53 122180619 Ki > 2000 nM T24983 CV1OA4 122180620 Ki > 3000 nM T24983 CYID81 122180621 Ki > 3000 nM T24983 CB91ZG 122180622 Ki > 1000 nM T24983 C1CIH2 122180623 Ki > 3000 nM T24983 C8YZ9Q 122180624 Ki > 20000 nM T24983 C9S3VH 122180625 Ki > 7000 nM T24983 CPRB82 122180954 Ki = 0.99 nM T24983 C08BVN 122180955 Ki = 2 nM T24983 CH9SX5 122180956 Ki = 10 nM T24983 CN7TP8 122181007 Ki = 3670 nM T24983 CCV9D5 122181326 Ki = 94 nM T24983 C91LDR 122181327 Ki = 36 nM T24983 CPW19F 122181328 Ki = 47 nM T24983 C5D1NC 122181329 Ki = 16 nM T24983 C05RGV 122181330 Ki = 34 nM T24983 C1KWI9 122181331 Ki = 31 nM T24983 CQ35XD 122181332 Ki = 40 nM T24983 C3XGN0 122181333 Ki = 1.4 nM T24983 C3BTQ7 122181334 Ki = 2370 nM T24983 CK5BP3 122189387 Ki = 37 nM T24983 C8JV3W 122189388 Ki = 130 nM T24983 CV1U4Q 122189389 Ki = 1400 nM T24983 C4PBA3 122189390 Ki = 3000 nM T24983 CD7UN3 122189391 Ki = 98 nM T24983 C14FCX 122189392 Ki = 180 nM T24983 C1NIK8 122189393 Ki = 42 nM T24983 C9KXH4 122189394 Ki = 76 nM T24983 CVJ3R4 122191605 Ki = 20 nM T24983 C2J4ZX 122191607 Ki = 0.72 nM T24983 C71KZQ 122205437 Ki = 188 nM T24983 C30ZRC 122205438 Ki = 72 nM T24983 CIAD86 126534204 Ki = 15848.93 nM T24983 C8K6JT 127027237 Ki = 59 nM T24983 CHY8I6 127027238 Ki = 730 nM T24983 C09YOS 127027905 Ki = 7.4 nM T24983 C3FAX7 127028181 Ki = 21 nM T24983 CU1HT7 127028182 Ki = 130 nM T24983 CMFY86 127028183 Ki = 73 nM T24983 CE9MN1 127028185 Ki = 3.3 nM T24983 C8MC1I 127028408 Ki = 1685 nM T24983 C9SC6E 127028505 Ki = 9.4 nM T24983 CNO74K 127029386 Ki = 13.1 nM T24983 CC7QN0 127029387 Ki = 10.8 nM T24983 C54KNW 127029388 Ki = 10.1 nM T24983 CBH17A 127029389 Ki = 26 nM T24983 C0MJ9C 127029390 Ki = 42 nM T24983 C3EQU4 127029391 Ki = 28 nM T24983 CX71NQ 127029995 Ki = 11.6 nM T24983 CB9MC5 127030606 Ki = 47 nM T24983 C8DPY4 127030612 Ki = 29 nM T24983 C9AC0T 127030909 Ki = 51 nM T24983 C5VP0F 127031201 Ki = 36 nM T24983 C76YBR 127031497 Ki = 27 nM T24983 CUV9A8 127031500 Ki = 35 nM T24983 C6T1PZ 127031508 IC50 = 62 nM T24983 CCOK40 127031513 Ki = 36 nM T24983 C5EU8Z 127031515 Ki = 14.3 nM T24983 CM5SK1 127031516 Ki = 10.4 nM T24983 C37NCK 127031518 Ki = 11.6 nM T24983 C12OBW 127031519 Ki = 16.1 nM T24983 CT86YX 127031829 Ki = 130 nM T24983 C4FU3T 127031830 Ki = 37 nM T24983 CP13VU 127031831 Ki = 5.4 nM T24983 CLIT39 127031832 Ki = 5.2 nM T24983 C0VSK2 127031833 Ki = 1060 nM T24983 CMHU98 127032082 Ki = 160 nM T24983 CS7W9I 127032083 Ki = 18.1 nM T24983 C3MGR1 127032084 Ki = 37 nM T24983 CW8LF2 127032085 Ki = 72 nM T24983 CMZ3A7 127032086 Ki = 47 nM T24983 CLIX68 127032383 Ki = 15.9 nM T24983 CD05QS 127032384 Ki = 2.2 nM T24983 CQ0ZT9 127035062 Ki = 853 nM T24983 CO53TS 127035828 Ki > 1000 nM T24983 CY7LP9 127035829 Ki > 1000 nM T24983 CR29BS 127035830 Ki > 1000 nM T24983 CU9C4S 127041952 Ki > 100000 nM T24983 C35GAL 127045853 Ki = 1400 nM T24983 C17LBT 127045854 Ki = 5400 nM T24983 CJ8GS7 127045855 Ki = 300 nM T24983 C2E1ZA 127046948 Ki = 9200 nM T24983 CTI5Z8 127046949 Ki = 900 nM T24983 C4D6BQ 127046950 Ki = 140 nM T24983 CM4CQ7 127046951 Ki = 1000 nM T24983 C29ERQ 127046952 Ki = 38 nM T24983 C78IFA 127047221 Ki = 240 nM T24983 CZL0U7 127047859 Ki = 55 nM T24983 CZ6XL5 127047996 Ki = 4.5 nM T24983 CC7BU0 127049059 Ki = 117.49 nM T24983 C42FHY 127049060 Ki = 1.549 nM T24983 CF2QY9 127049061 Ki = 671 nM T24983 CX53AC 127050632 Ki = 1512 nM T24983 CTL0S1 127051516 Ki = 131.83 nM T24983 CT9O7G 127051863 Ki = 229 nM T24983 C5ONG1 127051864 Ki = 432 nM T24983 CVQW26 127051865 Ki = 508 nM T24983 CSQ2N8 127052486 Ki = 831.76 nM T24983 C4YJ8H 127052487 Ki = 16 nM T24983 CT9RS4 127052488 Ki = 67.61 nM T24983 C14YJU 127052778 Ki = 1217 nM T24983 C1JAS7 127052779 Ki = 162.18 nM T24983 CLYU86 127053198 Ki = 42 nM T24983 C1Y9SB 127053214 Ki = 12.3 nM T24983 C89AWK 127053215 Ki = 44 nM T24983 CZRT07 127053217 Ki = 17.8 nM T24983 C8DV5I 127053218 Ki = 310 nM T24983 CC0NO4 127053219 Ki = 19.1 nM T24983 CA92IC 127053220 Ki = 150 nM T24983 CQ81AK 127053221 Ki = 16.2 nM T24983 CLE39U 127053222 Ki = 89 nM T24983 C10VDB 130431277 Ki = 316 nM T24983 CI1NF8 130431279 Ki = 2300 nM T24983 CS8O4E 130431287 Ki = 714 nM T24983 CR7T6X 130431290 Ki = 500 nM T24983 CU9XL0 130431303 Ki = 1960 nM T24983 C3MA6H 130431309 Ki > 10000 nM T24983 CDN26V 130431316 Ki = 5520 nM T24983 CL64UW 130431317 Ki = 2380 nM T24983 C8HE2O 130431318 Ki = 13900 nM T24983 C8ZHI7 130431325 Ki = 356 nM T24983 CEP1Q6 130431334 Ki = 305 nM T24983 CWT8I6 130431336 Ki = 503 nM T24983 CN70MW 130431337 Ki = 334 nM T24983 CIXV41 130431340 Ki = 529 nM T24983 C4GF1U 130431342 Ki = 5290 nM T24983 CWAC20 130431343 Ki = 819 nM T24983 C2WI5R 130431351 Ki = 1050 nM T24983 C50GOC 130442480 Ki = 6900 nM T24983 CM04RF 130442572 Ki = 6900 nM T24983 C1RI8Q 132060720 Ki = 904 nM T24983 CFXL21 132060812 Ki = 3.8 nM T24983 C7CSU4 132075278 Ki = 56 nM T24983 CAVB41 132584404 Ki > 10000 nM T24983 CBU81N 134149168 Ki > 10000 nM T24983 CRI9X8 135404757 Ki = 393 nM T24983 C4DZ5M 135418440 Ki = 21 nM T24983 CI4U9T 135442113 Ki = 89 nM T24983 CW60QI 135443755 Ki > 1000 nM T24983 CL87KM 135465626 Ki > 1000 nM T24983 CZXW36 135469096 Ki = 161 nM T24983 C21VFP 135470397 Ki > 1000 nM T24983 CINW45 135471592 Ki = 46 nM T24983 CRQE71 135479917 Ki > 1000 nM T24983 C8XYU4 135481864 Ki = 18 nM T24983 C1MTS9 135492584 Ki = 19 nM T24983 CW04LM 135493017 Ki > 1000 nM T24983 C5VXJ7 135493023 Ki > 1000 nM T24983 C3Q8AT 135501649 Ki = 510 nM T24983 C9EVN4 135501661 Ki > 1000 nM T24983 C7RQ2Y 135506137 Ki = 107 nM T24983 C0TY5Z 135514603 IC50 = 490 nM T24983 C2U1EP 135524323 Ki = 2.4 nM T24983 CZ52EH 135533255 Ki > 1000 nM T24983 C8AV4Z 135542446 Ki > 1000 nM T24983 C6LF4W 135545150 Ki = 341 nM T24983 CG95BM 135887931 Ki = 188 nM T24983 CQYI85 135887934 Ki = 50 nM T24983 C5W7CT 135887940 Ki = 3 nM T24983 C9Z6HJ 135921193 Ki = 3 nM T24983 CJEK87 135995891 Ki = 580 nM T24983 C89VLZ 136056636 Ki = 24 nM T24983 CZR53O 136072267 Ki = 52 nM T24983 C5CW3J 136094687 Ki = 125 nM T24983 CCEF36 136094866 Ki = 131 nM T24983 C96ZXY 136094867 Ki = 115 nM T24983 C4TF5O 137631542 Ki = 4.9 nM T24983 CN8BJ2 137632607 Ki = 210 nM T24983 C3R2LO 137632761 Ki = 11 nM T24983 C3PF9Z 137633454 Ki = 2100 nM T24983 COF9I6 137633705 Ki = 31 nM T24983 C8YM6U 137633863 Ki = 4.7 nM T24983 CN1I7A 137634153 Ki > 18000 nM T24983 C6FRJ5 137634397 Ki = 2.3 nM T24983 CPHI76 137635364 Ki = 160 nM T24983 C8ZFQ6 137635685 Ki = 55 nM T24983 C6QB9W 137635734 Ki = 28.84 nM T24983 CZ36LE 137636066 Ki = 60 nM T24983 CAL1W4 137636298 Ki = 6100 nM T24983 CX8O0V 137636308 Ki = 316.23 nM T24983 CAQ6I5 137636351 Ki = 30 nM T24983 C6GWQ3 137636460 Ki = 14 nM T24983 CQ20FO 137636498 Ki = 94 nM T24983 CZU6N5 137636581 Ki > 10000 nM T24983 C0YDQ5 137637428 Ki = 2600 nM T24983 C49VDK 137638973 Ki = 6.5 nM T24983 CA03VC 137639125 Ki = 51.29 nM T24983 C1HX3Z 137639304 Ki > 15000 nM T24983 CC16HE 137640152 Ki = 3200 nM T24983 CZP68A 137640189 Ki = 8.3 nM T24983 CZ4TA9 137640201 Ki = 1.259 nM T24983 CB2NO0 137640203 Ki = 11 nM T24983 CV49MZ 137640371 Ki = 7.9 nM T24983 CCU7L3 137640391 Ki = 17 nM T24983 CX4A3N 137640511 Ki = 257.04 nM T24983 C8IO0R 137640836 Ki = 270 nM T24983 C6PT7L 137642033 Ki = 880 nM T24983 C94WSH 137642380 Ki = 14 nM T24983 C4Q6ZM 137642607 Ki = 1.95 nM T24983 CAC6W0 137643122 Ki = 62 nM T24983 C71XIQ 137643132 Ki = 4700 nM T24983 CK51LB 137643309 Ki = 2.2 nM T24983 C3O0FX 137643951 Ki = 34 nM T24983 C34PUI 137644833 Ki = 19 nM T24983 C0KL6Q 137644962 Ki = 19.95 nM T24983 CVX6T1 137644966 Ki = 32 nM T24983 C4PV8U 137645196 Ki = 4900 nM T24983 CNH95X 137645574 Ki = 66 nM T24983 C3TP2G 137645830 Ki = 160 nM T24983 CG8P6I 137645938 Ki = 1.38 nM T24983 C96EAP 137646245 Ki = 36.31 nM T24983 CPI68E 137646281 EC50 = 359.1 nM T24983 CYH5U9 137647533 Ki = 5000 nM T24983 CSPE25 137649896 Ki = 2.8 nM T24983 CR3Z6M 137651073 Ki = 5.2 nM T24983 CW4T6D 137651322 Ki = 10 nM T24983 CMUT95 137651576 Ki = 95.5 nM T24983 C15YDU 137651936 Ki = 1.2 nM T24983 CX30HQ 137653096 Ki > 20000 nM T24983 CQ93DX 137653577 Ki = 8.8 nM T24983 C4C6EV 137653986 Ki = 440 nM T24983 COTX19 137654511 Ki = 560 nM T24983 CF5Y2A 137654675 Ki = 31 nM T24983 CLI4D8 137655029 Ki = 130 nM T24983 C7RW9H 137655451 Ki = 84 nM T24983 CJAZ13 137655556 Ki = 190 nM T24983 C6CA5H 137655594 Ki = 7600 nM T24983 CUC54G 137655636 Ki = 2.138 nM T24983 CDAN02 137655735 Ki = 8.1 nM T24983 CD16SQ 137655795 Ki = 300 nM T24983 CA7F5N 137657115 Ki = 7.8 nM T24983 CV2CR4 137657153 Ki = 54 nM T24983 CE0Y7P 137657322 Ki = 41 nM T24983 CRT86S 137657427 Ki = 75 nM T24983 CH76FP 137657951 Ki = 59 nM T24983 CEZ07P 137659303 Ki = 21 nM T24983 CP9AN6 137659990 Ki = 2 nM T24983 CP6US4 137660046 Ki = 4.8 nM T24983 C5V4DQ 137660707 Ki = 870 nM T24983 C42IDE 137660837 Ki = 1.5 nM T24983 CDA8V2 137661377 Ki = 5.248 nM T24983 CL58XS 145967572 Ki = 5.1 nM T24983 C58WSL 145967904 Ki = 114 nM T24983 CB1FD8 145968810 Ki = 54 nM T24983 C48XNG 145969667 Ki = 5.5 nM T24983 CNZY06 145969934 Ki = 11 nM T24983 C61MSO 145970938 Ki = 164 nM T24983 C1XF0I 145979855 Ki = 410 nM T24983 CO12QR 145979897 Ki = 1500 nM T24983 C87MSW 145980271 Ki = 10000 nM T24983 C8I7QL 145980875 Ki = 132 nM T24983 CP6DT9 145986441 Ki = 350 nM T24983 CNJH37 145986752 Ki = 459 nM T24983 CO4LK7 145988180 Ki = 14 nM T24983 CUGO10 145988693 Ki = 25 nM T24983 C4P6IC 145989012 Ki = 560 nM T24983 CLF26V 145990141 Ki = 140 nM T24983 CPW28Y 145990453 Ki = 170 nM T24983 CW87TZ 145991769 Ki = 150 nM T24983 CCP2U1 145992489 Ki = 1643 nM T24983 C74MRE 145993220 Ki = 1400 nM T24983 CRWE54 145993377 Ki = 720 nM T24983 CT29LQ 145993700 Ki = 660 nM T24983 C2H5AO 145993990 Ki = 95 nM T24983 CC2G1V 146025727 Ki = 4900 nM T24983 C6P3SR 153287553 Ki > 10000 nM T24983 CV9G7Z 153287572 Ki > 10000 nM T24983 CO85KL 153287574 Ki = 1995.26 nM T24983 CQ5WA9 155195311 Ki = 286 nM T24983 CUH20V 155195486 Ki = 2930 nM T24983 CG5NW0 155195487 Ki = 315 nM T24983 CJK6C0 155195495 Ki > 100000 nM T24983 C6ZV8B 155195496 Ki = 357 nM T24983 COJL79 155195501 Ki = 3220 nM T24983 C3MC0Q 155510756 Ki = 2.6 nM T24983 CTW28Q 155511803 Ki = 115.2 nM T24983 CJ96WB 155512259 Ki = 3.8 nM T24983 CQ83KZ 155512662 Ki = 806 nM T24983 C6XST7 155513053 Ki = 82.3 nM T24983 C0ZXT4 155513773 Ki = 3.4 nM T24983 CHXY56 155513802 Ki = 1298 nM T24983 CL5G9Q 155513837 Ki = 1047 nM T24983 CF6K8R 155514137 Ki = 46 nM T24983 CK9YN0 155514430 Ki = 322 nM T24983 CH34RK 155514798 Ki = 291.7 nM T24983 CV8F7A 155515301 Ki = 9772.37 nM T24983 C3XZM2 155515759 Ki = 33 nM T24983 CUE5J3 155515907 Ki = 1142 nM T24983 CM65NQ 155515931 Ki = 3.6 nM T24983 CUM2N4 155515982 Ki = 0.25 nM T24983 CV12SD 155516041 Ki = 676 nM T24983 CJ98ZK 155516236 Ki = 85.8 nM T24983 CH7N0C 155516494 Ki = 172.2 nM T24983 CQY58Z 155516873 Ki = 18 nM T24983 C9ZAW0 155517266 Ki = 215 nM T24983 C47LRQ 155518026 Ki = 16 nM T24983 CPER92 155519378 Ki = 4.4 nM T24983 CUSA24 155519891 Ki > 10000 nM T24983 C8IYD1 155520455 Ki = 179.2 nM T24983 C5DSE0 155520996 Ki = 100.8 nM T24983 CV7IG5 155522663 Ki = 326.1 nM T24983 CD59RE 155522719 Ki = 39290 nM T24983 C2H3JL 155523073 Ki = 384.6 nM T24983 CQA76T 155523112 Ki = 878 nM T24983 C3E9DJ 155523127 Ki = 2222 nM T24983 CG6Y4Z 155523515 Ki = 5.9 nM T24983 CVQ68Y 155523770 Ki = 844 nM T24983 COH1Q5 155524191 Ki = 813 nM T24983 CW7NT8 155524423 Ki = 1131 nM T24983 CQX27T 155525357 Ki = 1833 nM T24983 CT0NV4 155525431 Ki > 50000 nM T24983 CW65KS 155525705 Ki = 945 nM T24983 C9IW8F 155527714 Ki = 1.7 nM T24983 CUSG17 155529568 Ki = 36 nM T24983 C8U7QC 155529592 Ki = 4.6 nM T24983 C8WC5Y 155530733 Ki = 9 nM T24983 CDGX72 155530763 Ki = 76.4 nM T24983 C4VK0L 155531809 Ki = 44 nM T24983 C3R4YM 155532148 Ki = 1380.38 nM T24983 CKZ35G 155532475 Ki = 2884 nM T24983 C4LOR5 155532477 Ki = 988.6 nM T24983 CK9JP0 155532505 Ki = 3.3 nM T24983 CZA89B 155533824 Ki = 89.9 nM T24983 CQ12KS 155533996 Ki = 1585 nM T24983 C8AX5N 155534186 Ki = 2171 nM T24983 CZTX89 155534246 Ki = 2.9 nM T24983 CGZ5T8 155535272 Ki = 65.1 nM T24983 CHP2Z9 155535866 Ki = 510 nM T24983 CA01QX 155536022 Ki = 64 nM T24983 CB79ZW 155536080 Ki > 10000 nM T24983 CDEX60 155536720 Ki = 1.65 nM T24983 CY61EO 155536815 Ki = 110.4 nM T24983 CFCG03 155537361 Ki = 15 nM T24983 CVFD68 155537516 Ki = 575 nM T24983 C13CSU 155537907 Ki = 163 nM T24983 CP3WK6 155538028 Ki = 61 nM T24983 CFPT03 155538349 Ki = 14 nM T24983 C3DIY2 155539246 Ki = 132.8 nM T24983 CPV48W 155539557 Ki = 85.1 nM T24983 C9S2IA 155539605 Ki = 1283 nM T24983 CM9FI1 155542182 Ki = 15 nM T24983 CVK2M9 155543189 Ki = 1318 nM T24983 C4ANI0 155543691 Ki = 912 nM T24983 C08FTE 155544239 Ki = 2011 nM T24983 C7MCZ0 155546478 Ki = 376 nM T24983 C9D0GL 155547128 Ki = 20 nM T24983 C9GM0D 155548336 Ki = 28 nM T24983 CN6I4P 155550431 Ki = 1609 nM T24983 C6N9PG 155550640 Ki = 2171 nM T24983 CG7NR9 155550756 Ki = 2326 nM T24983 C82QWR 155551173 Ki = 553 nM T24983 CX8JA1 155552185 Ki = 0.55 nM T24983 CG70XQ 155552591 Ki = 1413 nM T24983 CB4F8Y 155552676 Ki = 962.3 nM T24983 C0DQ3Z 155552695 Ki = 400 nM T24983 CD5LC6 155554006 Ki = 575 nM T24983 CELU08 155555060 Ki = 5.9 nM T24983 C3UCM2 155557792 Ki = 275.42 nM T24983 C36SYJ 155558844 Ki = 220 nM T24983 CGBZ63 155559617 Ki = 0.55 nM T24983 C60GZE 155560295 Ki = 19 nM T24983 C7OZM6 155561446 Ki = 776 nM T24983 C75RMN 155561496 Ki = 6.5 nM T24983 CD2L9R 155561779 Ki = 12 nM T24983 CALB48 155561861 Ki > 10000 nM T24983 CF89GP 155562328 Ki = 6.2 nM T24983 C2Z0HB 155562353 Ki = 977.2 nM T24983 CRMC43 155562395 Ki = 6.87 nM T24983 C4IH5Z 155563301 Ki = 12.5 nM T24983 CAZL19 155563950 Ki = 21 nM T24983 CU7JG9 155564308 Ki = 2.6 nM T24983 C54WIE 155564667 Ki = 143 nM T24983 C0UN4V 155564747 Ki = 241 nM T24983 CMH8I1 155565768 Ki = 2073 nM T24983 CYIG07 155566058 Ki = 2.9 nM T24983 CRJG23 155566403 Ki = 9.7 nM T24983 CK20WA 155566662 Ki = 130 nM T24983 C6DPR8 155566974 Ki = 676 nM T24983 C95RAP 155567835 Ki = 501.2 nM T24983 C5A6YM 155567869 Ki = 1339 nM T24983 C8NO4X 155567971 Ki = 17 nM T24983 CQ5N6X 155568411 Ki = 5000 nM T24983 CV24CW 155568676 Ki = 671 nM T24983 C73ERT 155568786 Ki = 30 nM T24983 CKG5M1 155568867 EC50 = 1075 nM T24983 C42JKO 155569198 Ki = 851 nM T24983 CP9TR0 10324985 Ki = 8.5 nM T24983 C9J5HY 16105548 Ki = 28 nM T24983 C4ZD3A 16105549 Ki = 34 nM T24983 CB2VD8 44241743 Ki = 108 nM T24983 D00HUV 9881815 Ki = 51.6 nM T24983 D00NQV 5041 Ki = 0.33 nM T24983 D01ENR 2993172 Ki = 6484 nM T24983 D01GWH 44426510 Ki = 281 nM T24983 D01KIH 44323762 Ki = 47 nM T24983 D02NNS 9845181 Ki = 49 nM T24983 D02YDU 10420539 Ki > 20000 nM T24983 D03DET 10287730 Ki < 10000 nM T24983 D03GES 9995378 Ki = 130 nM T24983 D03JEW 44431485 Ki = 181 nM T24983 D03JOS 233952 Ki = 8 nM T24983 D03KUH 57267 Ki = 70.4 nM T24983 D03PYX 1219 Ki = 148 nM T24983 D03VPS 16094676 EC50 = 89 nM T24983 D04CPW 25139331 Ki = 6100 nM T24983 D04JUJ 54456 Ki = 6400 nM T24983 D04PBA 10015867 Ki > 400 nM T24983 D05BCJ 2779264 Ki = 1100 nM T24983 D05EQG 5265 Ki = 0.2 nM T24983 D05HMW 10705550 Ki > 20000 nM T24983 D05LJF 44431481 Ki = 34 nM T24983 D05QJK 9816808 Ki = 315.5 nM T24983 D05UUW 210956 Ki = 2 nM T24983 D05XNR 10034684 Ki = 500 nM T24983 D05ZUX 44207909 Ki >= 1000 nM T24983 D06AIQ 107995 Ki = 570 nM T24983 D06BWZ 68678 Ki > 10000 nM T24983 D06FUV 5311189 Ki = 16 nM T24983 D06NTB 30438 Ki = 570 nM T24983 D06VDN 443391 IC50 > 1000 nM T24983 D06WLB 9838216 Ki = 230.2 nM T24983 D07GQP 11477180 Ki = 375 nM T24983 D07LRJ 5312149 Ki = 130 nM T24983 D07QMR 44426502 Ki = 362 nM T24983 D07RYR 44396235 Ki = 1428 nM T24983 D07UUQ 15508240 Ki = 940 nM T24983 D07VBS 10425450 EC50 = 2.7 nM T24983 D08QPU 72737723 Ki = 36 nM T24983 D08TCX 11437461 Ki > 10000 nM T24983 D09CVG 449126 Ki > 3300 nM T24983 D09FTZ 10564794 Ki = 16000 nM T24983 D09FZD 35296170 Ki = 139 nM T24983 D09RPR 16737207 Ki > 10000 nM T24983 D09WBJ 10336538 Ki = 2.188 nM T24983 D0A2BE 2780 Ki = 3.2 nM T24983 D0AW4X 44431465 Ki = 66 nM T24983 D0AX0K 5615 IC50 = 8 nM T24983 D0B0UZ 9861462 EC50 = 2.4 nM T24983 D0B9DR 15508243 Ki = 1500 nM T24983 D0C0LG 44426508 Ki = 29 nM T24983 D0C0UM 10775317 Ki > 20000 nM T24983 D0C5RZ 5610 Ki > 35000 nM T24983 D0E1PL 9865384 Ki = 2000 nM T24983 D0E1RX 11335419 Ki = 1261 nM T24983 D0E3AL 56597938 Ki = 76 nM T24983 D0F0IA 11301655 Ki = 1.5 nM T24983 D0FF6S 16038374 IC50 > 10000 nM T24983 D0FK5Z 35295787 Ki = 230 nM T24983 D0G0IQ 3802 Ki = 36 nM T24983 D0G2CP 10404144 Ki = 2 nM T24983 D0G8CV 9954003 Ki = 1.585 nM T24983 D0G8VU 3645619 Ki = 2.3 nM T24983 D0H2IT 9928335 Ki = 42 nM T24983 D0H2WQ 54562 EC50 = 1.4 nM T24983 D0I8MP 16725931 Ki = 36 nM T24983 D0IU8V 9903877 Ki = 10 nM T24983 D0J1HP 10378389 Ki = 11.75 nM T24983 D0K3UL 9796720 Ki = 3.6 nM T24983 D0L5MW 181743 Ki = 262 nM T24983 D0L7OM 6917970 Ki = 3748 nM T24983 D0M2BB 25333445 Ki = 20 nM T24983 D0M2ZE 6604756 Ki = 48 nM T24983 D0M3PV 133633 Ki = 220 nM T24983 D0O1PM 4420454 Ki = 22 nM T24983 D0O3GF 1220 Ki > 1515 nM T24983 D0O4BC 11776546 Ki = 80.6 nM T24983 D0O9BZ 2728532 Ki = 14.7 nM T24983 D0OG0R 10337743 IC50 > 5000 nM T24983 D0P0IX 16104 Ki = 16 nM T24983 D0P7OB 9798466 Ki = 7.8 nM T24983 D0Q2GP 10381810 Ki = 23 nM T24983 D0Q4DP 6603897 Ki = 0.51 nM T24983 D0Q5IP 10851078 Ki = 25 nM T24983 D0R8UU 44396220 Ki = 4476 nM T24983 D0S1XN 44323962 Ki = 2.6 nM T24983 D0S7WZ 5119 Ki > 933 nM T24983 D0SL4Q 46190878 Ki = 2511.89 nM T24983 D0T1TU 68950 Ki > 10000 nM T24983 D0T2RY 9948320 Ki = 11 nM T24983 D0TU5W 44323978 Ki = 1.7 nM T24983 D0V4NW 25139332 Ki = 1400 nM T24983 D0V5OY 16725912 Ki = 11 nM T24983 D0WD6J 10357869 Ki = 63 nM T24983 D0WU9R 133008 Ki = 2.5 nM T24983 D0X1QW 122334 Ki = 117 nM T97035 D03UOT 785 IC50 = 4400000 nM T97035 D08HVR 6047 IC50 = 8400000 nM T97035 D04PBH 5280804 IC50 > 50000 nM T97035 D0U3EP 445154 IC50 = 250000 nM T97035 D09SWE 31244 IC50 = 320000 nM T97035 D0NH9P 135 IC50 = 9350 nM T97035 C4N9ZB 240 IC50 = 820000 nM T97035 CVAK03 326 IC50 = 50000 nM T97035 C12TIO 6998 IC50 = 3300000 nM T97035 CT7K0H 69600 IC50 = 30000 nM T97035 C7P3UR 69975 Ki = 128000 nM T97035 CC2SV8 100528 IC50 > 50000 nM T97035 CD1JI7 124052 IC50 = 90 nM T97035 COZ0S4 158516 EC50 = 90000 nM T97035 CYWS98 185848 IC50 = 8000 nM T97035 CV5XP0 440936 IC50 = 30260 nM T97035 CTLB85 480774 IC50 = 7500 nM T97035 C1MQG9 480859 IC50 = 177 nM T97035 C0MZK5 480860 IC50 = 154 nM T97035 C9OI2P 1268251 IC50 > 250000 nM T97035 CFB78O 1551008 IC50 > 250000 nM T97035 CC40IA 1909086 IC50 > 250000 nM T97035 CG5B4N 4564493 IC50 = 50000 nM T97035 CVK40B 5280704 IC50 > 50000 nM T97035 CL1MR9 5281254 IC50 = 38400 nM T97035 CY4H3A 5317025 IC50 > 50000 nM T97035 CI58XK 5319562 IC50 = 30000 nM T97035 CO4EU9 5321954 IC50 > 50000 nM T97035 CK7WJ9 5354004 IC50 > 100000 nM T97035 CWS5X0 5481970 IC50 = 23 nM T97035 CZP6R5 5488795 IC50 > 50000 nM T97035 CRU8Z2 6604874 IC50 > 100000 nM T97035 CH8N0L 9851181 IC50 > 50000 nM T97035 C47UMD 10149024 IC50 = 2300 nM T97035 C4YPN1 10371980 IC50 = 330 nM T97035 CX36QB 10439562 IC50 = 240 nM T97035 C8G1SE 11579720 IC50 = 31700 nM T97035 C8X7MR 11623165 IC50 = 38000 nM T97035 CEH78Q 11844492 IC50 = 2210000 nM T97035 C30RKD 11844493 IC50 = 70000 nM T97035 CPFW43 11844494 IC50 = 140000 nM T97035 C84BVJ 13943263 IC50 = 54640 nM T97035 CD17LS 14482777 IC50 > 50000 nM T97035 CIJS40 21626605 IC50 = 102390 nM T97035 C1P2GB 21630099 IC50 = 48920 nM T97035 CHQO58 44139786 IC50 > 250000 nM T97035 CPWI05 44274763 IC50 = 23210 nM T97035 CLGD42 44274791 IC50 = 3030 nM T97035 C0NZ1Q 44274946 IC50 = 14510 nM T97035 CN7J6B 44274954 IC50 = 2000 nM T97035 CVO2R6 44274955 IC50 = 60 nM T97035 C5E4SJ 44274988 IC50 = 2390 nM T97035 CHMF54 44274989 IC50 = 8000 nM T97035 CF6PY7 44275023 IC50 = 16660 nM T97035 CQ4Z5R 44328350 IC50 = 2130 nM T97035 CG86MP 44328543 IC50 = 6170 nM T97035 C8ON7H 44328544 IC50 = 4480 nM T97035 CV0E5S 44328644 IC50 = 390 nM T97035 CD9E3Y 44328645 IC50 = 780 nM T97035 CF4Y2U 44328721 IC50 = 2180 nM T97035 C5AIR7 44406314 IC50 > 10000000 nM T97035 CJK74L 44406702 IC50 = 92250 nM T97035 CQ62YP 44419358 IC50 > 100000 nM T97035 CY7Q3X 44419359 IC50 > 100000 nM T97035 CB78SU 44419360 IC50 > 100000 nM T97035 CYA04R 44419367 IC50 > 100000 nM T97035 CJU0H5 44559660 IC50 = 333000 nM T97035 C4ZGX5 44579614 IC50 = 1600 nM T97035 CTM59H 44579615 IC50 = 430 nM T97035 CQ6U4N 44579616 IC50 = 730 nM T97035 C74FMO 44583889 IC50 = 450000 nM T97035 CW9QP8 44584115 IC50 = 85010 nM T97035 CK4D9A 46864286 Ki = 350 nM T97035 C5Q0HJ 46864287 IC50 = 30000 nM T97035 CR13OY 49800619 IC50 = 9100 nM T97035 CMX4N3 52916198 IC50 = 770 nM T97035 CC48ZA 52916199 IC50 = 680 nM T97035 C98SIU 52916200 IC50 = 830 nM T97035 C6C5WM 56657821 IC50 = 700 nM T97035 C5PF2S 56668245 IC50 = 15350 nM T97035 CVM26Y 66563419 IC50 = 417000 nM T97035 CCZ6P5 71768558 IC50 = 4560 nM T97035 CJM24N 71768559 IC50 = 1510 nM T97035 CPY3E1 71768560 IC50 = 3830 nM T97035 C4T7SH 71768561 IC50 = 1980 nM T97035 C8WQY9 71768562 IC50 = 4130 nM T97035 C1R7EH 71769044 IC50 = 2300 nM T97035 C1XR4F 71769045 IC50 = 4720 nM T97035 C69FHY 72163243 IC50 = 42800 nM T97035 CI8DV1 72163245 IC50 = 12600 nM T97035 C8D1ME 72946266 IC50 = 1720 nM T97035 CCU72B 122191010 IC50 = 2170 nM T97035 C19NRX 122191011 IC50 = 1780 nM T97035 C9MVJ7 127045527 IC50 = 1950 nM T97035 CN7Q2K 132504095 IC50 = 2800 nM T97035 C5DHW3 134153783 IC50 = 34000 nM T97035 CMFA91 134852570 IC50 = 290000 nM T97035 C2WA4Z 137638552 IC50 = 5100 nM T97035 C8R0CZ 145956637 IC50 = 45300 nM T97035 CU27XS 145986129 IC50 = 170 nM T97035 CEI03S 155511909 IC50 = 4620 nM T97035 CI4HT1 155515316 IC50 = 4770 nM T97035 CWTC68 155527800 IC50 > 50000 nM T97035 CLV74A 155530485 IC50 > 50000 nM T97035 CE96SD 155532290 IC50 = 8970 nM T97035 CFY0Q5 155532440 IC50 = 7890 nM T97035 C95ECX 155534997 IC50 > 50000 nM T97035 CE78RC 155550073 IC50 > 50000 nM T97035 C90TBX 155568103 IC50 > 50000 nM T97035 D02CFH 676454 IC50 = 1800 nM T97035 D02JEZ 5281426 IC50 = 420000 nM T97035 D03QNS 5393176 IC50 > 10000000 nM T97035 D04ZQC 24180539 IC50 = 15210 nM T97035 D06ZRX 5281717 IC50 = 12700 nM T97035 D07DAP 24849532 IC50 = 370 nM T97035 D07EGB 3610 IC50 = 560 nM T97035 D07HYL 16126762 IC50 = 1600 nM T97035 D07RGP 44406305 IC50 = 13950 nM T97035 D09XKH 10356745 IC50 = 980 nM T97035 D09YJS 24180556 IC50 = 14500 nM T97035 D0A6ZK 80297 IC50 > 1000000 nM T97035 D0AU0M 637542 IC50 = 3000 nM T97035 D0BH2T 10107266 IC50 = 70 nM T97035 D0BH6B 13844658 IC50 > 50000 nM T97035 D0DQ2G 16043 IC50 = 54200 nM T97035 D0F3CO 3840 IC50 = 7400 nM T97035 D0G3TK 5280863 IC50 = 1000 nM T97035 D0H4YW 3611 IC50 = 8980 nM T97035 D0IO0I 6474893 IC50 > 250000 nM T97035 D0J6RQ 6437306 IC50 = 79050 nM T97035 D0M2EN 205912 IC50 = 21000 nM T97035 D0U8JC 9862769 IC50 = 80 nM T97035 D0Z1XR 12649 IC50 = 1150 nM T97035 D0ZR4M 5276405 IC50 = 4930 nM T72849 D0RA5Q 72172 IC50 = 50000 nM T72849 CDBF98 281242 Ki > 250000 nM T72849 C6L1VE 1551321 Ki = 249000 nM T72849 C4BKQ3 4798291 Ki = 3800 nM T72849 CUX8S7 7197248 IC50 = 9200 nM T72849 CN5H0B 10970861 Ki = 6470 nM T72849 C5OPG0 11127644 Ki = 26900 nM T72849 C10KPB 11142955 Ki = 19100 nM T72849 CF19DX 13509139 Ki > 250000 nM T72849 C4Y1HP 15849848 Ki > 250000 nM T72849 CVRO49 25760265 IC50 = 14400 nM T72849 CX18KT 44447089 Ki = 6270 nM T72849 C1CXM0 45292546 IC50 = 3000 nM T72849 CO34LD 45464518 IC50 = 20200 nM T72849 CN53IO 53792079 Ki > 250000 nM T72849 C7P2UD 71817806 IC50 = 95500 nM T72849 CMQN63 71817809 IC50 = 2000 nM T72849 C1N7QD 71817963 IC50 = 7700 nM T72849 C74CNV 72193911 IC50 = 33 nM T72849 CI4Q9X 73437636 IC50 = 7400 nM T72849 CU8WB9 73437637 IC50 = 8600 nM T72849 CRU02V 74766022 Ki = 5550 nM T72849 CX5CN1 76401637 IC50 = 6900 nM T72849 CJ2UC1 85470733 IC50 = 8200 nM T72849 CRA08X 85470742 IC50 = 15200 nM T72849 C05HWU 86140993 Ki > 250000 nM T72849 CR0PF5 86222557 IC50 = 32600 nM T72849 CF35LZ 87495845 Ki > 250000 nM T72849 CVS60Z 118720629 Ki = 31600 nM T72849 C4VWL9 118720630 Ki = 530 nM T72849 C71CKB 118720631 Ki = 87100 nM T72849 CCQ74S 118720632 Ki = 11300 nM T72849 C8JDP5 118720633 Ki = 991 nM T72849 CE9X4G 118720634 Ki = 12300 nM T72849 CW87DK 118720635 Ki = 2540 nM T72849 CKIF61 118720636 Ki > 250000 nM T72849 CJ6MY3 118720637 Ki = 18600 nM T72849 CP5V7M 118720638 Ki = 3730 nM T72849 CB67XZ 118734161 IC50 > 100000 nM T72849 C67EIN 118734163 IC50 > 100000 nM T72849 C5HV4G 118734165 IC50 > 100000 nM T72849 CR02XN 118734172 IC50 > 100000 nM T72849 CYQ61P 118734173 IC50 > 100000 nM T72849 CG1NJ3 118734176 IC50 = 6800 nM T72849 CTL4C9 118734177 IC50 = 18300 nM T72849 C1UWG8 118734178 IC50 = 42000 nM T72849 C24VOF 118734181 IC50 = 110000 nM T72849 C3KJR9 118734182 IC50 > 100000 nM T72849 CMWH70 118734252 IC50 = 9800 nM T72849 CS1R6T 118734253 IC50 = 12100 nM T72849 CK3NV4 118734254 IC50 > 100000 nM T72849 C4VK6O 118734255 IC50 = 38400 nM T72849 C7AH4D 118734256 IC50 > 100000 nM T72849 CZ97HL 118734258 IC50 > 100000 nM T72849 C1DKP8 118734259 IC50 = 920 nM T72849 CET0D8 118734260 IC50 = 3600 nM T72849 C4N7KF 118734261 IC50 = 10700 nM T72849 C3PL1T 118734263 IC50 = 9600 nM T72849 C3OS1H 118734264 IC50 = 1200 nM T72849 C9NWC0 118734265 IC50 > 100000 nM T72849 C6IB5P 118734270 IC50 > 100000 nM T72849 CI9RT3 118734273 IC50 > 100000 nM T72849 CK32TS 118734274 IC50 = 35000 nM T72849 C96PKA 118734278 IC50 = 9400 nM T72849 C4AL9Z 118734279 IC50 = 13400 nM T72849 C71TGN 118734280 IC50 = 12000 nM T72849 CIZ3Q6 118734282 IC50 = 16700 nM T72849 CJ64ZC 118734283 IC50 = 1100 nM T72849 C1K7AN 118734284 IC50 = 19500 nM T72849 C6XY9M 118734285 IC50 > 100000 nM T72849 CO4F3Y 118734287 IC50 = 800 nM T72849 C9CN6S 118734288 IC50 = 8900 nM T72849 CN7SR4 118734290 IC50 > 100000 nM T72849 CKST54 118734292 IC50 > 100000 nM T72849 C9XDY5 118734293 IC50 = 2500 nM T72849 C01PYL 118734294 IC50 = 2800 nM T72849 C4ZPC8 118734296 IC50 = 2600 nM T72849 CJ40TN 118734297 IC50 = 38200 nM T72849 C7FMV5 126456392 Ki = 3500 nM T72849 C7UJ4W 127043855 IC50 = 520 nM T72849 CW0FZ2 127044995 Ki = 1520 nM T72849 C06JOP 127044996 Ki = 4940 nM T72849 CM0VT4 127048200 Ki > 250000 nM T72849 CTL4Z8 127048201 Ki > 250000 nM T72849 CBQ4S3 127048202 Ki > 250000 nM T72849 CC96VU 127048834 Ki > 250000 nM T72849 CTY5D4 127049157 Ki > 250000 nM T72849 CF3HO2 127049196 Ki > 250000 nM T72849 C03XKF 127049491 Ki > 250000 nM T72849 CFW6M1 127049492 Ki > 250000 nM T72849 CL6D0Z 127049497 Ki > 250000 nM T72849 C4I1RH 127049824 Ki > 250000 nM T72849 C2A1MZ 127050130 Ki > 250000 nM T72849 CA4MP3 127050430 Ki > 250000 nM T72849 CJT5R9 127050433 Ki > 250000 nM T72849 C0N2LE 127050745 Ki > 250000 nM T72849 C9GBD2 127051304 Ki > 250000 nM T72849 CLK50R 127051701 Ki > 250000 nM T72849 C2BUZ7 127051959 Ki > 250000 nM T72849 CK81ME 127051999 Ki > 250000 nM T72849 CAC25R 127052273 Ki > 250000 nM T72849 C3FMN7 127052612 Ki > 250000 nM T72849 CHA9Q6 127052870 Ki > 250000 nM T72849 CJM96B 127053163 Ki > 250000 nM T72849 C3TK6A 135547192 IC50 = 43000 nM T72849 C8QO7V 135554374 IC50 = 18000 nM T72849 C7H3GR 135641933 IC50 = 27000 nM T72849 CXLS30 137633011 IC50 = 1969 nM T72849 CMC5E8 137634250 IC50 = 126 nM T72849 CER06G 137637900 IC50 = 25111 nM T72849 C97XKO 137638141 IC50 = 31212 nM T72849 CMTG53 137639983 IC50 = 7473 nM T72849 CH6DQ2 137640549 IC50 > 100000 nM T72849 C9SWV7 137640590 IC50 = 726 nM T72849 CG0ED2 137641900 IC50 = 949 nM T72849 C3SP9K 137642894 IC50 = 21229 nM T72849 C1U3ZM 137642974 IC50 = 3093 nM T72849 CYN9Z5 137646376 IC50 = 143 nM T72849 CDU93R 137646849 IC50 = 178 nM T72849 C96EWT 137647165 IC50 = 682 nM T72849 CJM57W 137648545 IC50 = 102 nM T72849 CC9T7O 137650040 IC50 = 65 nM T72849 CN9F2A 137650752 IC50 = 2650 nM T72849 CB9VI7 137652734 IC50 = 2518 nM T72849 CSM3V5 137653412 IC50 > 100000 nM T72849 CVI87E 137654495 IC50 > 35000 nM T72849 C8DV5C 137655020 IC50 = 2660 nM T72849 C2RIG6 137655030 IC50 = 33 nM T72849 CMT56C 137655972 IC50 = 2087 nM T72849 C13POW 137656080 IC50 = 27008 nM T72849 CCTK37 137657323 IC50 = 71 nM T72849 C4VS2D 137658289 IC50 = 98 nM T72849 CKHE71 137659752 IC50 = 48 nM T72849 C0ID7T 137660529 IC50 = 43 nM T72849 C8E6UD 137661774 IC50 = 340 nM T72849 CV2U0Z 137662110 IC50 = 155 nM T72849 CB1J0U 145994843 Ki = 17500 nM T72849 C94BDA 155510769 IC50 = 124000 nM T72849 CJMO47 155512116 Ki = 44000 nM T72849 CYE4R8 155512732 IC50 = 170000 nM T72849 CK9D4I 155512960 IC50 = 150000 nM T72849 C0CYS7 155515712 IC50 = 115000 nM T72849 C7VYT6 155517480 IC50 = 165000 nM T72849 CIH73R 155523459 Ki = 4700 nM T72849 CD0F5Z 155524591 IC50 = 6900 nM T72849 CGOU03 155531602 IC50 > 10000 nM T72849 CY1MF9 155534671 IC50 > 200000 nM T72849 C8E6QH 155538090 Ki = 23400 nM T72849 CZG6O5 155539882 IC50 = 135000 nM T72849 C8XYO7 155545269 Ki = 10900 nM T72849 C8R0JW 155547335 IC50 = 1995.26 nM T72849 CF35ER 155548478 IC50 = 3694 nM T72849 CQM59I 155550629 IC50 > 10000 nM T72849 COR09W 155554600 Ki = 18500 nM T72849 CRU97I 155558560 IC50 > 100000 nM T72849 CRVJ23 155564248 IC50 > 100000 nM T72849 CU0W9L 155566815 IC50 = 3600 nM T72849 CHEX85 445715 Ki = 5080 nM T72849 D02MNM 71817810 IC50 = 2600 nM T94912 D0G2XE 6918468 IC50 = 15.85 nM T94912 CU96IB 131577 Ki = 150000 nM T94912 CVJ46C 223995 IC50 > 100 ug.mL-1 T94912 C0LQG3 234070 IC50 > 100 ug.mL-1 T94912 CU3I9S 234079 IC50 > 100 ug.mL-1 T94912 CQ23YV 235632 IC50 > 60000 nM T94912 CQX4M9 265219 IC50 = 200 nM T94912 C7REB9 408239 IC50 > 50 ug.mL-1 T94912 CQJP09 1250946 EC50 > 60000 nM T94912 C03YNW 1351023 IC50 = 14600 nM T94912 C84SMK 1379975 IC50 = 8700 nM T94912 C39LPI 3196682 IC50 = 125.89 nM T94912 COT07B 3453336 IC50 = 59 nM T94912 C7MGQ3 5773323 IC50 = 12 ug.mL-1 T94912 CJ20TS 5909556 IC50 = 30 ug.mL-1 T94912 C2V4XW 9989013 EC50 = 48000 nM T94912 C9DA2N 10010954 IC50 = 490 nM T94912 CEM2F0 10011515 EC50 = 15800 nM T94912 CKI8Q7 10011643 EC50 = 2500 nM T94912 CR5SZ2 10057217 EC50 = 1200 nM T94912 CQ5IL1 10102925 EC50 = 4000 nM T94912 CXM30U 10260801 EC50 = 224000 nM T94912 C2L1OB 10328378 IC50 = 1995.26 nM T94912 CJ8L9B 10351296 EC50 = 300 nM T94912 C3J7VK 10351393 EC50 = 2100 nM T94912 CA17CG 10374110 EC50 = 5600 nM T94912 CMN41C 10374115 Ki = 390 nM T94912 C48BDO 10396578 EC50 = 4000 nM T94912 CM2C6S 10418298 IC50 = 360 nM T94912 CJFK61 10418799 EC50 = 215000 nM T94912 C3RMH6 10418817 EC50 = 19500 nM T94912 C0V2GR 10418881 EC50 = 22000 nM T94912 CUT40G 10441364 EC50 = 50000 nM T94912 CX0LR4 10441383 EC50 = 5000 nM T94912 CF3EV2 10463109 IC50 = 55000 nM T94912 CSO5E8 10464003 EC50 = 2300 nM T94912 CW8D9N 10464012 EC50 = 70000 nM T94912 C3OD5Q 10464120 EC50 = 500000 nM T94912 CRK13Y 10486513 IC50 = 4700 nM T94912 C7XFQ8 10510226 IC50 = 2600 nM T94912 C3MW1N 10557548 IC50 = 144000 nM T94912 CO7FW9 10557793 IC50 = 2951.21 nM T94912 CFY13C 10616508 IC50 = 2000 nM T94912 C0VUX7 10629679 IC50 = 5888.44 nM T94912 CP6KR5 10653515 IC50 = 51000 nM T94912 C1ONR5 10724409 IC50 = 700 nM T94912 CM7AT6 10724498 IC50 > 42657.95 nM T94912 C29SYI 10795799 IC50 = 12 nM T94912 CWA0K3 10796341 IC50 = 4570.88 nM T94912 CE3C2X 10819181 IC50 < 1000000 nM T94912 C6XU3O 10819260 IC50 = 9000 nM T94912 C5LQT4 10819534 IC50 = 500 nM T94912 CRA0F6 10843359 IC50 = 1949.84 nM T94912 CW1S3T 11766790 EC50 = 2000 nM T94912 C1OIT7 11803878 IC50 = 3548.13 nM T94912 CFUP74 11857314 IC50 = 90 nM T94912 C9T6HG 12253728 IC50 > 100000 nM T94912 CI0W3Z 12253756 IC50 = 30000 nM T94912 CCK8Z0 12473171 EC50 > 60000 nM T94912 C51CXK 14588192 IC50 = 1.7 ug.mL-1 T94912 C4NZ3E 15133383 IC50 = 2 ug.mL-1 T94912 COIX70 15133384 IC50 = 18 ug.mL-1 T94912 C2PY5T 15133385 IC50 > 50 ug.mL-1 T94912 C68FSN 15133387 IC50 > 100 ug.mL-1 T94912 CDXI20 15133388 IC50 > 50 ug.mL-1 T94912 C4UK1G 15133390 IC50 = 9 ug.mL-1 T94912 C9YG1I 15133392 IC50 > 50 ug.mL-1 T94912 CCB82L 15133393 IC50 > 100 ug.mL-1 T94912 C49TDH 15133396 IC50 > 100 ug.mL-1 T94912 CONB25 15133397 IC50 > 50 ug.mL-1 T94912 CM48AT 15133398 IC50 > 100 ug.mL-1 T94912 CLR8T7 15133399 IC50 = 8 ug.mL-1 T94912 CFBH58 15133400 IC50 = 30 ug.mL-1 T94912 C4ZHX7 15133401 IC50 = 30 ug.mL-1 T94912 C34QHN 15133402 IC50 = 4 ug.mL-1 T94912 CY6BQ4 15133403 IC50 = 7 ug.mL-1 T94912 C1RS9Y 15133405 IC50 > 100 ug.mL-1 T94912 CU54OK 15133406 IC50 > 100 ug.mL-1 T94912 C7NZE4 15133407 IC50 > 100 ug.mL-1 T94912 C8I5AS 15725946 Ki = 210000 nM T94912 C5PIR8 15725947 Ki = 25000 nM T94912 CGV6N1 15725948 Ki = 10000 nM T94912 CCF07N 15725949 Ki = 750000 nM T94912 CQJB30 15725952 Ki = 2900 nM T94912 CI9T5B 15725956 Ki = 2000 nM T94912 CK37JY 15725957 Ki = 1600 nM T94912 CW9YH0 15725958 Ki = 5300 nM T94912 C2Y3PS 17615045 IC50 = 44500 nM T94912 C1ZIJ0 24894075 IC50 = 7 nM T94912 CHR1V9 24970311 IC50 = 1 nM T94912 CLBN94 25010731 Ki = 8.9 nM T94912 CBJ5U6 25108851 IC50 = 51 nM T94912 CI0P1S 25109118 IC50 = 18 nM T94912 CY4IA6 25109473 IC50 = 26 nM T94912 CMF20W 25109614 IC50 = 25 nM T94912 C2QVM4 25109748 IC50 = 22 nM T94912 C9P8SK 25110775 IC50 = 125 nM T94912 C3Y7OS 25110776 IC50 = 90 nM T94912 CC0D4T 25191127 IC50 = 3200 nM T94912 CGO76M 25191129 IC50 = 3500 nM T94912 CN07LF 25191131 Ki = 3700 nM T94912 CH67ZI 25191132 IC50 = 4900 nM T94912 CDJY09 25191261 IC50 = 2600 nM T94912 CLTQ86 25191262 IC50 = 5000 nM T94912 C7ITF9 25191265 Ki = 370 nM T94912 C93JHW 25191266 IC50 = 6200 nM T94912 C6V1YK 25191388 Ki = 680 nM T94912 CG0WP7 25191514 IC50 = 6200 nM T94912 C28CUR 25191639 IC50 = 22 nM T94912 CCB8K5 25191640 IC50 = 26 nM T94912 C1FUH4 25191762 Ki = 21 nM T94912 C2XA8H 25191763 IC50 = 37 nM T94912 CV0HO8 25191764 IC50 = 53 nM T94912 CKR41V 25191765 IC50 = 67 nM T94912 C6A9NV 25191766 Ki = 13 nM T94912 CK2Z4S 25191896 IC50 = 82 nM T94912 C42QJX 25191897 Ki = 10 nM T94912 C9AUZ1 25191898 IC50 = 110 nM T94912 C5UC2L 25191899 Ki = 180 nM T94912 C3N6MS 25191900 IC50 = 120 nM T94912 CRJ5S2 25191901 IC50 = 130 nM T94912 CR01FX 25192049 Ki = 7.3 nM T94912 CDY74P 25192050 IC50 = 170 nM T94912 CB5DG7 25192196 IC50 = 180 nM T94912 CI1YP8 25192198 IC50 = 220 nM T94912 CUG5S4 25192200 Ki = 9.7 nM T94912 CE1FC6 25192335 IC50 = 270 nM T94912 C2DB6J 25192336 IC50 = 290 nM T94912 C57AGT 25192337 IC50 = 340 nM T94912 CR42YT 25192338 IC50 = 350 nM T94912 CD4J3C 25192339 Ki = 35 nM T94912 CUM4B7 25192488 IC50 = 410 nM T94912 CYS9R5 25192489 IC50 = 420 nM T94912 C6YI9W 25192490 IC50 = 430 nM T94912 C0HR8P 25192491 IC50 = 530 nM T94912 C2J9GL 25192493 IC50 = 560 nM T94912 CR0DC8 25192633 Ki = 86 nM T94912 CVHX47 25192634 IC50 = 690 nM T94912 CM3A6J 25192635 IC50 = 730 nM T94912 CM60NU 25192636 IC50 = 790 nM T94912 CJ3N7G 25192638 IC50 = 840 nM T94912 CATD54 25192764 IC50 = 880 nM T94912 CNU76Z 25192765 IC50 = 910 nM T94912 CCG2W3 25192766 IC50 = 950 nM T94912 C9T0DF 25192769 IC50 = 1400 nM T94912 C8ZQI3 25192896 IC50 = 1400 nM T94912 C3TG7E 25192897 IC50 = 1500 nM T94912 C1WAL2 25192898 IC50 = 1500 nM T94912 CAW5M1 25192901 IC50 = 1700 nM T94912 C25YCL 25193028 IC50 = 1700 nM T94912 CV04ES 25193029 Ki = 1200 nM T94912 C8SUH0 25193031 Ki = 180 nM T94912 C5TNI1 25193057 IC50 = 22 nM T94912 C8Q7VT 25193171 IC50 = 2400 nM T94912 CN24JP 25193172 IC50 = 2400 nM T94912 C2IP0H 25193174 IC50 = 2500 nM T94912 CB8ZC4 25193175 IC50 = 2600 nM T94912 C2L8UV 44301802 IC50 = 3090.3 nM T94912 CJ3R4O 44301857 IC50 > 16982.44 nM T94912 CIQ6K0 44301938 IC50 = 3200 nM T94912 CA96CM 44301960 IC50 = 16000 nM T94912 C6SI5F 44301966 IC50 = 41000 nM T94912 CC28KW 44301970 IC50 > 56.23 nM T94912 CWQG56 44301971 IC50 = 9500 nM T94912 CUT45G 44301983 IC50 > 269.15 nM T94912 C9VEY4 44301984 IC50 = 10000 nM T94912 CU58SH 44301986 IC50 = 300 nM T94912 CQ4N1X 44302015 IC50 = 3800 nM T94912 C56WNL 44302230 IC50 = 300 nM T94912 C4KS0O 44302231 IC50 = 8100 nM T94912 C2YPH6 44305324 Ki = 300000 nM T94912 CI0J4B 44305325 EC50 = 1.3 nM T94912 CO52KR 44305625 Ki = 100000 nM T94912 C5HD0K 44308822 IC50 = 4000 nM T94912 CI89BA 44342908 IC50 = 1800 nM T94912 CY5QI1 44347020 EC50 = 500000 nM T94912 CLB4Y1 44353001 Ki = 2100 nM T94912 C9Q5PJ 44353002 Ki = 260 nM T94912 CT89UX 44353003 Ki = 220 nM T94912 C4VP3O 44353014 Ki = 810 nM T94912 CFG6T2 44353020 Ki = 4400 nM T94912 C2BVM0 44353031 Ki = 36000 nM T94912 C7WVA2 44353032 Ki = 31000 nM T94912 CPJH61 44353033 Ki = 13000 nM T94912 CGCD74 44353083 Ki = 79000 nM T94912 C21JOP 44353179 Ki = 20000 nM T94912 C79ULO 44353181 Ki = 180000 nM T94912 CPJE52 44383008 IC50 = 8000 nM T94912 C4LIR7 44383043 IC50 = 50000 nM T94912 CE2F7V 44383126 IC50 = 4000 nM T94912 CY59VJ 44383127 IC50 = 6000 nM T94912 C17BQM 44383144 IC50 = 25000 nM T94912 CS92WK 44383275 IC50 = 4000 nM T94912 C1CM4J 44383378 IC50 = 7500 nM T94912 CPAU45 44383557 IC50 = 54000 nM T94912 CV13QW 44383558 IC50 = 8000 nM T94912 C6OXP9 44383561 IC50 = 9000 nM T94912 CA8MJ7 44383980 IC50 = 1000 nM T94912 C3XK4L 44384139 IC50 = 1000 nM T94912 CQ76HO 44384193 IC50 = 3000 nM T94912 CCD43W 44384304 IC50 = 30000 nM T94912 CDUN52 44384305 IC50 = 9000 nM T94912 C12REV 44384385 IC50 = 9000 nM T94912 CANV51 44384438 IC50 = 4500 nM T94912 CL7QI6 44416525 IC50 = 45 nM T94912 CKX67V 44416526 IC50 = 146 nM T94912 C8HC6X 44416527 IC50 = 300 nM T94912 C3OU9B 44416533 IC50 = 107 nM T94912 C8TJ0K 44416733 IC50 = 19 nM T94912 C3JK6V 44417104 IC50 = 535 nM T94912 CXW34I 44417113 IC50 = 190 nM T94912 C2HU1Z 44417114 IC50 = 463 nM T94912 CF2B7K 44417116 IC50 = 31 nM T94912 CEI6S5 44417117 IC50 = 63 nM T94912 C9DZ7B 44417118 IC50 = 27 nM T94912 CI37CH 44417122 IC50 = 116 nM T94912 CD0N8O 44417123 IC50 = 60 nM T94912 CFQ1X6 44417124 IC50 = 71 nM T94912 CDV29A 44417129 IC50 = 8700 nM T94912 CCFZ48 44417130 IC50 = 18 nM T94912 CR7BY2 44417153 IC50 = 50 nM T94912 CE3Q0O 44417158 IC50 = 54 nM T94912 C0JZ4C 44417159 IC50 = 57 nM T94912 CFED63 44417160 IC50 = 38 nM T94912 C0ID8W 44417199 IC50 = 23000 nM T94912 C1W7JC 44417200 IC50 = 25 nM T94912 CV58SG 44417205 IC50 = 100000 nM T94912 C8KD3J 44417206 IC50 = 6900 nM T94912 CD29CK 44417227 IC50 = 76 nM T94912 C58PXI 44448386 IC50 = 1900 nM T94912 CSI3H4 44448415 IC50 = 820 nM T94912 C8FM7R 44450395 IC50 > 10000 nM T94912 CAD15P 44450396 IC50 > 10000 nM T94912 CX54WI 44450403 IC50 > 10000 nM T94912 CKBH61 44450404 IC50 > 10000 nM T94912 C2XK3U 44450405 IC50 > 10000 nM T94912 C0G2DZ 44450406 IC50 > 10000 nM T94912 CT06GI 44450415 Ki = 8300 nM T94912 CR1FM5 44450416 IC50 > 10000 nM T94912 C3FX7L 44450417 IC50 > 10000 nM T94912 CY51GX 44450426 IC50 > 10000 nM T94912 CF17EP 44450439 IC50 > 10000 nM T94912 CLV38B 44450446 IC50 > 10000 nM T94912 CSX9T4 44450456 IC50 > 10000 nM T94912 CID60S 44450457 IC50 > 10000 nM T94912 CV2P8R 44450458 IC50 > 10000 nM T94912 CN6XM9 44450467 IC50 > 10000 nM T94912 CE06GZ 44450488 IC50 > 10000 nM T94912 CM0SP7 44567879 IC50 > 10000 nM T94912 CIJ0N7 44567913 IC50 > 10000 nM T94912 CV32CF 44567970 IC50 > 10000 nM T94912 CP4I5X 44567971 IC50 = 7400 nM T94912 CBN84U 44568046 IC50 > 10000 nM T94912 CR5L6E 44568047 IC50 > 10000 nM T94912 C4NP2D 44568090 IC50 = 380 nM T94912 CYFO65 44568091 IC50 > 10000 nM T94912 CNG7Z5 44568130 IC50 > 10000 nM T94912 CWDA52 44568131 IC50 > 10000 nM T94912 C86IZV 44568165 IC50 > 10000 nM T94912 CVY97F 44568166 IC50 > 10000 nM T94912 CXV3I6 44581449 IC50 = 3 nM T94912 CKI6S0 44581481 IC50 > 1000 nM T94912 C73AWH 44581482 IC50 = 15 nM T94912 C37UCL 44581483 IC50 = 350 nM T94912 C2L0EX 44581484 IC50 = 8 nM T94912 C2JS7Q 44581545 IC50 = 12 nM T94912 CT8Z4K 44581546 IC50 = 45 nM T94912 CAF9Z3 44581547 IC50 = 25 nM T94912 CZ4I3G 44581572 IC50 > 1000 nM T94912 CMP1H4 44581573 IC50 = 200 nM T94912 COT17R 44581574 IC50 = 500 nM T94912 C9FVK0 44581575 IC50 = 90 nM T94912 CA3Y0D 44581615 IC50 = 500 nM T94912 C8D0GS 44581616 IC50 = 47 nM T94912 CD7FM9 44581617 IC50 > 1000 nM T94912 CLSO84 44581650 IC50 > 1000 nM T94912 CG4FT8 44581651 IC50 > 1000 nM T94912 CT5F9X 44581652 IC50 = 790 nM T94912 C8VT9H 44581653 IC50 = 325 nM T94912 CXS0Z7 44589629 IC50 = 1000 nM T94912 CC7Z5W 44589630 IC50 = 330 nM T94912 C01SWN 44589666 IC50 = 200 nM T94912 CBY26Z 44589667 IC50 > 1000 nM T94912 C6QWD4 44589668 IC50 = 350 nM T94912 CAP4K2 44589669 IC50 = 70 nM T94912 CN9L6Q 44589704 IC50 = 75 nM T94912 C8X5PR 44589705 IC50 > 1000 nM T94912 CI4NQ2 44589706 IC50 > 1000 nM T94912 CG9WX7 44589707 IC50 = 175 nM T94912 CSX1G9 44589742 IC50 = 370 nM T94912 CO93SH 44589743 IC50 = 5 nM T94912 C69RYZ 44589744 IC50 > 1000 nM T94912 CDI78W 44589781 IC50 > 1000 nM T94912 C2OAD8 44589782 IC50 = 1000 nM T94912 C28QPO 44589783 IC50 = 80 nM T94912 CE0JI6 44589784 IC50 > 1000 nM T94912 CNVA28 44589817 IC50 = 835 nM T94912 CDHK69 44589818 IC50 = 175 nM T94912 CG9V3Y 44589819 IC50 = 1.5 nM T94912 C86FTU 44589820 IC50 = 18 nM T94912 CQ54PU 44589862 IC50 = 400 nM T94912 CSOE13 44589863 IC50 = 110 nM T94912 C96FOQ 44589864 IC50 = 300 nM T94912 CASQ04 44589865 IC50 = 35 nM T94912 C9D6YM 44589919 IC50 > 1000 nM T94912 CHB0V5 44589920 IC50 = 395 nM T94912 C2SB3O 44589921 IC50 = 90 nM T94912 CY8L7K 44589922 IC50 = 435 nM T94912 CPW64I 44589976 IC50 = 5 nM T94912 C7PUR0 44589977 IC50 = 89 nM T94912 C0N1KC 44589978 IC50 = 290 nM T94912 C7ER1D 44590340 IC50 = 1000 nM T94912 CR9MF1 44590341 EC50 = 123.03 nM T94912 CTV9J3 44590401 IC50 > 10000 nM T94912 CP30EL 44590402 IC50 > 10000 nM T94912 CS58YP 44590403 IC50 = 794.33 nM T94912 CA49GO 44590404 IC50 > 10000 nM T94912 C3RH8X 44590445 IC50 = 63.1 nM T94912 CP9SU5 44590446 IC50 > 100 nM T94912 CXOC39 44590447 IC50 = 19.95 nM T94912 CVL1S9 44590448 IC50 = 39.81 nM T94912 CWVR62 44590515 IC50 = 100 nM T94912 CJ17UF 44590516 IC50 = 199.53 nM T94912 CZ93YT 44590517 IC50 = 316.23 nM T94912 CA6BM0 44590518 IC50 = 3162.28 nM T94912 C4GR0W 44593654 IC50 = 31 nM T94912 C0PQA1 46225376 EC50 > 60000 nM T94912 C2O1HF 46225392 EC50 > 60000 nM T94912 C2KJV1 46225393 IC50 > 60000 nM T94912 CK8QW4 46225413 IC50 = 400 nM T94912 CW78DI 49799080 IC50 = 501.19 nM T94912 C8PH3O 49799081 IC50 = 1995.26 nM T94912 CO48HR 49799082 IC50 = 29000 nM T94912 C2ANS9 73345497 Ki = 200 nM T94912 CX2Z7N 73354472 Ki = 150000 nM T94912 CX3SC2 100972207 IC50 = 4786.3 nM T94912 CM20FH 100972208 IC50 = 794.33 nM T94912 CM31ZT 118719096 Ki = 600000 nM T94912 C60AYU 118719108 IC50 = 3000 nM T94912 CA2P9V 118719109 IC50 > 173.78 nM T94912 C2N9JO 118719110 IC50 = 1200 nM T94912 D00HAJ 73347136 IC50 = 39 nM T94912 D03QAN 71166 IC50 = 3.3 ug.mL-1 T94912 D03TBA 10020451 IC50 = 800 nM T94912 D04JXA 5311122 IC50 = 3 nM T94912 D09MAZ 46897162 IC50 > 5000 nM T94912 D0J3FH 10218379 Ki = 15.2 nM T31956 CKWA31 125415 Ki = 2300 nM T31956 CXT3Z6 168101 Ki = 2400 nM T31956 CW10CK 439518 Ki = 8000 nM T31956 C30OXI 9990739 Ki = 840 nM T31956 CAN9H3 10251613 Ki = 13 nM T31956 CFW39X 10261412 Ki = 980 nM T31956 CQV19H 10262161 Ki = 510 nM T31956 CM6DT8 10352382 Ki = 390 nM T31956 CVD02L 10397127 Ki = 130 nM T31956 C24AMZ 10651513 Ki = 150 nM T31956 CN5H0B 10970861 Ki = 67 nM T31956 CYR08N 19366756 Ki = 17200 nM T31956 CF4VL0 21120524 Ki = 140 nM T31956 CUBV96 44276209 Ki = 870 nM T31956 C34DUK 44276215 Ki = 1900 nM T31956 C9CUN1 44276216 Ki = 2400 nM T31956 C32JVB 44276289 Ki = 2000 nM T31956 C79TMD 44276303 Ki > 3000 nM T31956 C4JB1Z 44276401 Ki > 3000 nM T31956 CQX6J3 44276410 Ki = 2800 nM T31956 CV5MC9 44276625 Ki = 2700 nM T31956 CHP16B 44276842 Ki = 2200 nM T31956 CHVC96 44331549 Ki = 4100 nM T31956 CE5X0Q 44331641 Ki = 1600 nM T31956 CT05NF 44331710 Ki = 370 nM T31956 CGF91D 44331721 Ki = 280 nM T31956 CMD6C1 44331731 Ki = 2000 nM T31956 CSEP-73 44331732 Ki = 290 nM T31956 CZDN46 44331761 Ki = 870 nM T31956 C1G4ED 44331762 Ki = 3500 nM T31956 CHY17G 44365802 Ki = 51 nM T31956 CRGI20 44365950 Ki = 80 nM T31956 CH1LQ0 145974448 Ki = 40000 nM T31956 CL8NR9 145975342 Ki = 130 nM T31956 CSQK47 10531941 Ki = 27 nM T31956 CQ7Z6E 10628244 Ki = 9.3 nM T31956 CQBZ03 10650722 Ki = 292 nM T31956 C90UTY 10745654 Ki = 14.7 nM T31956 CA02QN 10841584 Ki = 4.3 nM T31956 COHR67 11802605 Ki = 73.3 nM T31956 CR0M5B 44365322 Ki = 910 nM T31956 CI79UQ 44365364 Ki = 240 nM T31956 C1Z6AM 44365366 Ki = 3.83 nM T31956 C87WDI 44365382 Ki = 110 nM T31956 CS9OG6 44365505 Ki = 12 nM T31956 CDV05R 44365525 Ki = 3.2 nM T31956 C4TK3N 44365528 Ki = 53 nM T31956 CP17OQ 44365564 Ki = 83.3 nM T31956 C1P7ZR 44365567 Ki = 3.6 nM T31956 C4UP8J 44365591 Ki = 283 nM T31956 C1G6QO 44365607 Ki = 5.36 nM T31956 CWN1H8 44365642 Ki = 4200 nM T31956 CY4GA8 44365645 Ki = 145 nM T31956 CKY54U 44365647 Ki = 1200 nM T31956 CR3VQ7 44365649 Ki = 40 nM T31956 CUD15T 44365873 Ki = 20 nM T31956 CTRJ90 44365886 Ki = 50 nM T31956 C2R1PL 44365889 Ki = 470 nM T31956 C26YMC 44365892 Ki = 15 nM T31956 C10JTG 44365896 Ki = 267 nM T31956 CC4JW5 44365908 Ki = 3.56 nM T31956 C6Y1EN 44365910 Ki = 13 nM T31956 C7K3DX 44365936 Ki = 16 nM T31956 D0B9ZE 44365325 Ki = 0.873 nM T78992 D0K8KX 5280343 IC50 = 4230 nM T78992 D03HUX 49792852 IC50 > 10000 nM T78992 D0E3TC 44259 IC50 > 10000 nM T78992 D0O0LS 25141092 IC50 > 10000 nM T78992 D0P1CV 46191454 IC50 > 10000 nM T78992 D0Q9UX 16718576 IC50 = 1065 nM T78992 C8IAR2 5281657 IC50 > 100000 nM T78992 CI68PW 5283685 IC50 > 100000 nM T78992 CXK0S6 5283727 IC50 > 100000 nM T78992 C4G9WR 9547398 IC50 > 100000 nM T78992 C76CUP 9547698 IC50 > 100000 nM T78992 CR8DA1 10024683 IC50 > 100000 nM T78992 CLA93G 10047202 IC50 > 100000 nM T78992 C3LCH5 10047545 IC50 > 100000 nM T78992 C4CP7K 10423452 IC50 = 67800 nM T78992 C7HBP6 10429593 IC50 > 10000 nM T78992 C83QWV 10714343 IC50 = 7720 nM T78992 C8G5WP 11210533 IC50 = 1850 nM T78992 C7YG1N 24759534 IC50 = 8800 nM T78992 C5YW7P 24825755 IC50 = 1664 nM T78992 C4EG8R 24993189 IC50 > 10000 nM T78992 CNG96H 25210579 IC50 > 10000 nM T78992 CU3RF1 45139989 IC50 > 10000 nM T78992 CQGZ06 45139991 IC50 > 10000 nM T78992 C7ON5A 46233287 IC50 > 10000 nM T78992 CF91RS 49843531 IC50 > 10000 nM T78992 CBC62W 50899254 IC50 = 595 nM T78992 C2Y6QS 50938552 IC50 > 10000 nM T78992 C9NYP4 51036677 IC50 > 10000 nM T78992 C4WRY3 51037112 IC50 > 10000 nM T78992 CRI28Z 51037948 IC50 > 10000 nM T78992 CE1ZK6 54759168 IC50 > 10000 nM T78992 C9ZFS1 54764923 IC50 > 100000 nM T78992 CBZ8T4 56657856 IC50 = 336 nM T78992 CYPL60 56675140 IC50 > 10000 nM T78992 CXJ63M 59603829 IC50 = 5900 nM T78992 CQEU96 59603842 IC50 = 2600 nM T78992 CV63UL 67240318 IC50 > 10000 nM T78992 C5DGR9 69036886 IC50 = 10000 nM T78992 CCN01X 71547862 IC50 > 10000 nM T78992 C3UC9H 73891099 IC50 = 520 nM T78992 CV8QX0 76310169 IC50 > 30000 nM T78992 CA5L4W 76324771 IC50 > 30000 nM T78992 C9GO0P 76328313 IC50 = 13600 nM T78992 C39FTZ 76335685 IC50 > 100000 nM T78992 C1HW4B 89735655 IC50 = 17000 nM T78992 CY0UC4 90645194 IC50 > 10000 nM T78992 CY7BI2 118706214 IC50 > 10000 nM T78992 C2AN7T 134611886 IC50 > 100000 nM T78992 CHA4N2 136013680 IC50 > 10 nM T78992 C1YUD0 136219394 IC50 > 10 nM T78992 CIU8W3 136254389 IC50 > 10 nM T78992 C2MD1Q 155513187 IC50 > 10000 nM T78992 D03DZO 11715767 IC50 > 10000 nM T78992 D08HFG 24809764 IC50 > 10000 nM T78992 D09HVH 135566652 IC50 > 10 nM T78992 D0C1DQ 6490494 IC50 = 59800 nM T78992 D0T8NU 16757525 IC50 > 4000 nM T35527 D02HWP 2722 IC50 = 1900 nM T35527 D09JUG 60490 IC50 = 55000 nM T35527 D0K8KX 5280343 IC50 = 440 nM T35527 D0DK4I 4534 IC50 = 180 nM T35527 CD6W3K 6618 IC50 = 10000 nM T35527 CUO98K 7808 IC50 > 100000 nM T35527 CFQ35W 11563 IC50 > 100000 nM T35527 C4T5QC 11847 IC50 > 100000 nM T35527 C0NHG2 12005 IC50 > 100000 nM T35527 CP1V2F 68523 IC50 > 100000 nM T35527 C9CLG6 70119 IC50 > 100000 nM T35527 CY0AL9 72279 IC50 > 100000 nM T35527 C6CLP5 80801 IC50 = 5000 nM T35527 C0JLT2 125100 IC50 = 3800 nM T35527 CDV60U 125101 IC50 = 17000 nM T35527 C1H8NR 155248 IC50 = 210 nM T35527 CDN7P9 156398 IC50 = 7600 nM T35527 C7FL5H 173513 IC50 = 1600 nM T35527 C13WSH 195771 IC50 = 410 nM T35527 C0SMD7 339231 IC50 = 410 nM T35527 C05QAO 353995 IC50 > 100000 nM T35527 C9XA6R 356358 IC50 = 70000 nM T35527 CF2YR7 356359 IC50 = 26000 nM T35527 CS0DT8 476858 IC50 = 42000 nM T35527 C0A8BP 487903 IC50 > 40000 nM T35527 C97DNA 637177 IC50 = 39000 nM T35527 CV97HM 663693 IC50 > 100000 nM T35527 CJ2L1C 688659 IC50 > 100000 nM T35527 CCY5N0 727302 IC50 > 100000 nM T35527 CBM8Y0 771546 IC50 > 100000 nM T35527 CPM12N 775994 IC50 > 50000 nM T35527 CIHN92 785627 IC50 = 30700 nM T35527 C0BD2V 801015 IC50 > 200000 nM T35527 CVF50J 836505 IC50 > 100000 nM T35527 CF2MW6 854652 IC50 = 12300 nM T35527 C9QO5R 883201 IC50 > 100000 nM T35527 COE63U 889785 IC50 > 100000 nM T35527 CIEY41 1072992 IC50 > 100000 nM T35527 C38XKW 1079725 IC50 > 40000 nM T35527 C3Q2CD 1079726 IC50 > 40000 nM T35527 CA1TU5 1079729 IC50 = 5100 nM T35527 C1S4HO 1079730 IC50 = 22000 nM T35527 CFO62A 1082938 IC50 > 200000 nM T35527 CG6KC7 1095055 IC50 > 200000 nM T35527 C81MSC 1141363 IC50 > 100000 nM T35527 CWE1Y9 1304061 IC50 > 100000 nM T35527 CUD6L7 1325172 IC50 > 200000 nM T35527 CW1JO4 1346428 IC50 > 200000 nM T35527 C8Z2PM 1743704 IC50 > 200000 nM T35527 CC25XB 1998811 IC50 > 100000 nM T35527 CAJ10O 2192753 IC50 > 500000 nM T35527 CD0X5M 2920571 IC50 = 1000 nM T35527 CU16KY 2920793 IC50 = 1000 nM T35527 CIB83N 2921053 IC50 = 3000 nM T35527 C4UJQ1 2921716 IC50 = 800 nM T35527 CJ4B3F 2921923 IC50 = 1200 nM T35527 C92GBS 2931181 IC50 > 100000 nM T35527 CZ02OG 2933060 IC50 > 200000 nM T35527 C1OTU9 3136123 IC50 = 3400 nM T35527 C5DB7U 3136132 IC50 > 150000 nM T35527 C3G9QL 3136134 IC50 = 380 nM T35527 CF3NM8 5280701 IC50 = 1000 nM T35527 C0D3PO 5281671 IC50 = 100000 nM T35527 C17CBF 5281812 IC50 > 100000 nM T35527 C2NKF5 5283162 IC50 = 8000 nM T35527 C0WXP5 5284649 IC50 = 8700 nM T35527 C6IVR9 5317326 IC50 = 14000 nM T35527 C6D3GZ 5393151 IC50 > 100000 nM T35527 CV56UY 5407860 IC50 = 6400 nM T35527 CV0B7K 5481241 IC50 = 1600 nM T35527 C7P4ZA 5713107 IC50 > 100000 nM T35527 CQZ8U3 6446027 IC50 > 100000 nM T35527 CS4MF3 9586795 IC50 > 200000 nM T35527 C4T9ES 10020717 IC50 5000 nM T35527 C20LUF 10072931 IC50 = 430 nM T35527 CF8Y2Q 10340455 IC50 = 360 nM T35527 CZ8B7D 10348509 IC50 = 6200 nM T35527 C4NXL5 10554258 IC50 = 12000 nM T35527 CV0RN7 10905139 IC50 = 26000 nM T35527 C13UBC 10914853 IC50 = 780 nM T35527 C0OX8Y 10936155 IC50 = 620 nM T35527 CWN43C 10937563 IC50 = 360 nM T35527 C1R5SB 10955008 IC50 > 100000 nM T35527 CHT16X 11019578 IC50 > 10000 nM T35527 C9IH6W 11041857 IC50 > 100000 nM T35527 C7IGY5 11142891 IC50 = 3100 nM T35527 CA4TQ6 11248759 IC50 > 3000 nM T35527 C6RG5B 11466350 IC50 = 9700 nM T35527 CCX16G 11532986 IC50 > 10000 nM T35527 C8PJ6B 11677372 IC50 > 10000 nM T35527 C6GVK4 14983007 IC50 > 100000 nM T35527 CNHZ34 15628203 IC50 = 15000 nM T35527 C9WDR1 21270142 IC50 = 780 nM T35527 CBJ87P 21270161 IC50 = 3600 nM T35527 CT94AD 21270186 IC50 = 11000 nM T35527 CXQW24 21831939 IC50 > 100000 nM T35527 CEFB61 23093378 IC50 > 100000 nM T35527 CBV19H 23425708 IC50 > 200000 nM T35527 C4YJM0 24721289 IC50 > 100000 nM T35527 C9DO6A 24825393 IC50 = 1070 nM T35527 CK7M8I 24825399 IC50 > 10000 nM T35527 CFN79S 24825402 IC50 > 10000 nM T35527 CQK5S6 24825412 IC50 > 10000 nM T35527 CBY15M 33845371 IC50 = 480 nM T35527 CN31MU 44142338 IC50 > 75000 nM T35527 CL0G1O 44142340 IC50 > 75000 nM T35527 CB24IA 44142341 IC50 > 50000 nM T35527 C3PZ1K 44142342 IC50 = 1200 nM T35527 C4NTK0 44142343 IC50 = 1600 nM T35527 C78WJH 44142344 IC50 > 150000 nM T35527 CB7C0P 44142345 IC50 = 2600 nM T35527 CWC96M 44142346 IC50 = 3000 nM T35527 CPX7M3 44142347 IC50 > 75000 nM T35527 C5IMG1 44142348 IC50 > 75000 nM T35527 CY6N1P 44142350 IC50 = 5000 nM T35527 CX50WK 44142351 IC50 = 2000 nM T35527 C37APD 44323089 IC50 = 2200 nM T35527 C0BRV6 44396187 IC50 = 5100 nM T35527 COH1B3 44436892 IC50 = 4900 nM T35527 CXF24P 44437715 IC50 > 100000 nM T35527 CI7NA6 44437716 IC50 > 100000 nM T35527 C8GU3K 44437717 IC50 > 100000 nM T35527 C5I9VM 44437718 IC50 > 100000 nM T35527 C3VE4H 44437719 IC50 > 100000 nM T35527 CXK29W 44437720 IC50 > 100000 nM T35527 C9B0CX 44437721 IC50 > 100000 nM T35527 CV6W4R 44437722 IC50 > 100000 nM T35527 C7RWS3 44437723 IC50 > 100000 nM T35527 CN40UP 44437724 IC50 > 100000 nM T35527 CVBQ79 44437725 IC50 > 100000 nM T35527 C40KOY 44437726 IC50 > 100000 nM T35527 CJ1DA0 44437727 IC50 > 100000 nM T35527 C4KD8Z 44437728 IC50 > 100000 nM T35527 CWMX75 44437729 IC50 > 100000 nM T35527 C2WSB6 44437731 IC50 = 5800 nM T35527 CQT74A 44437732 IC50 = 14000 nM T35527 C2XZV9 44460112 IC50 > 100000 nM T35527 CNK7B4 44460114 IC50 > 100000 nM T35527 CG1I0J 44460122 IC50 > 100000 nM T35527 C7W1HI 44460123 IC50 > 100000 nM T35527 C4B0ZM 44460128 IC50 > 100000 nM T35527 C9OR2U 44460130 IC50 > 100000 nM T35527 CX4GJ6 44460139 IC50 > 100000 nM T35527 CDAY05 44460167 IC50 > 75000 nM T35527 CQ85JS 44460168 IC50 = 3500 nM T35527 CEF14Q 44460169 IC50 > 50000 nM T35527 C5H9MT 44460172 IC50 = 2000 nM T35527 C5DY0N 44460173 IC50 = 14000 nM T35527 C5J7ED 44460174 IC50 = 2000 nM T35527 C2XWI4 44460175 IC50 = 430 nM T35527 CM85EO 44460178 IC50 > 150000 nM T35527 C9G6EW 44460179 IC50 > 75000 nM T35527 CGR42M 44460180 IC50 > 75000 nM T35527 C0QD8O 44557858 IC50 > 150000 nM T35527 CJX28F 46213934 IC50 > 10000 nM T35527 CM17VT 46926342 IC50 > 25000 nM T35527 CW8L7D 46926343 IC50 > 25000 nM T35527 C2PL3G 46927848 IC50 > 10000 nM T35527 CB7XA0 49788946 IC50 > 100000 nM T35527 C4O0QK 49821278 IC50 > 20000 nM T35527 C64KTI 51042131 IC50 > 10000 nM T35527 C5GRB6 54754354 IC50 > 10000 nM T35527 C3YM2E 54754518 IC50 > 10000 nM T35527 CN3F5O 56641761 IC50 > 10000 nM T35527 C7ZI3H 56642018 IC50 > 10000 nM T35527 CU1G5A 56642290 IC50 > 10000 nM T35527 C0SM7Z 56642536 IC50 > 10000 nM T35527 C6TLW3 56642537 IC50 > 10000 nM T35527 C8M1ZL 70701358 IC50 = 3700 nM T35527 CRI98P 70701360 IC50 = 1300 nM T35527 CMS29P 70701361 IC50 = 2500 nM T35527 C79FQU 70701362 IC50 > 40000 nM T35527 CI8NG5 70701363 IC50 = 5600 nM T35527 C74ZIE 70701364 IC50 = 11000 nM T35527 C32ORS 70701366 IC50 = 6300 nM T35527 CJLA95 70701367 IC50 = 2200 nM T35527 CN4XW9 70701368 IC50 = 2300 nM T35527 CGKU94 70701370 IC50 > 40000 nM T35527 CKD43S 70701371 IC50 = 4200 nM T35527 C1NBV9 70701372 IC50 = 350 nM T35527 CN7G0U 70701373 IC50 > 40000 nM T35527 CCH5F9 70701374 IC50 = 700 nM T35527 CPHC34 70701376 IC50 = 2200 nM T35527 CQON52 70701377 IC50 = 6200 nM T35527 CA76MQ 70701378 IC50 = 570 nM T35527 C2LCZ6 70701381 IC50 = 4500 nM T35527 CPI2U9 70701382 IC50 = 12000 nM T35527 C07DVY 70701383 IC50 > 40000 nM T35527 C92ZAQ 70701385 IC50 = 240 nM T35527 CRJ4S1 70701387 IC50 = 500 nM T35527 CZ90TO 70701389 IC50 = 4500 nM T35527 CYC5H3 70701390 IC50 = 480 nM T35527 CSB8U0 70701391 IC50 > 40000 nM T35527 CO7QX0 70701393 IC50 = 510 nM T35527 C7R2VZ 70701396 IC50 = 2300 nM T35527 CCP7U1 70701397 IC50 = 3500 nM T35527 C62NYQ 70701398 IC50 = 7000 nM T35527 C6K5YI 70701399 IC50 > 40000 nM T35527 CE1VL6 70701400 IC50 > 40000 nM T35527 CB17XD 70701401 IC50 > 40000 nM T35527 C71SMJ 70701406 IC50 = 1600 nM T35527 C7CY2A 70701407 IC50 > 40000 nM T35527 CK3O6T 70701411 IC50 = 1300 nM T35527 CGYX64 70701412 IC50 = 330 nM T35527 CFR72B 70701413 IC50 = 1300 nM T35527 CBA34S 70701414 IC50 = 11000 nM T35527 CLUJ38 70701415 IC50 > 40000 nM T35527 COU80L 70701416 IC50 = 1400 nM T35527 C82OSZ 70701419 IC50 > 40000 nM T35527 CC86DV 70701421 IC50 = 6300 nM T35527 C9UVN4 70701422 IC50 = 19000 nM T35527 C09PML 70701424 IC50 > 40000 nM T35527 CF1HR0 70701425 IC50 = 13000 nM T35527 CGWB74 70701426 IC50 = 340 nM T35527 C3LG4O 70701428 IC50 = 5300 nM T35527 CO5BE9 70701429 IC50 > 40000 nM T35527 C3BU8G 70701430 IC50 = 2900 nM T35527 CT4IL7 70701432 Ki = 530 nM T35527 C8C7KL 70701433 IC50 = 5000 nM T35527 CUW26F 70701435 IC50 = 2700 nM T35527 CZ40JM 70701440 IC50 = 3000 nM T35527 C2J5QD 70701441 IC50 > 40000 nM T35527 CFB82A 70701443 IC50 = 5000 nM T35527 C21SFN 70701445 IC50 = 1700 nM T35527 CSP6X9 70701446 IC50 > 40000 nM T35527 CR48TX 70701447 IC50 > 40000 nM T35527 CTZ59M 71307312 IC50 = 1300 nM T35527 C2OZ9H 72375189 IC50 > 10000 nM T35527 CF7HU4 76314061 IC50 > 40000 nM T35527 CV0BO9 76317616 IC50 = 180 nM T35527 CW5Y2X 76317617 IC50 = 1100 nM T35527 CIM93K 76321347 IC50 = 390 nM T35527 CIK5A0 76321348 IC50 = 260 nM T35527 CO7KA5 76321349 IC50 = 220 nM T35527 CHG2K7 76324948 IC50 = 4000 nM T35527 CO8FC6 76332190 IC50 > 40000 nM T35527 CN6AE5 76332191 IC50 = 160 nM T35527 CIS0R8 76335724 IC50 > 10000 nM T35527 CP13GH 76335828 IC50 = 3800 nM T35527 CN31IU 76335829 IC50 = 760 nM T35527 CL3XS0 81689867 IC50 > 10000 nM T35527 CSB0M9 135494223 IC50 = 7300 nM T35527 CST9B8 136244569 IC50 = 7700 nM T35527 D00YEV 5281605 IC50 = 860 nM T35527 D01KKU 5281894 IC50 > 100000 nM T35527 D03YMX 11093078 IC50 = 6000 nM T35527 D04JWS 324974 IC50 = 150 nM T35527 D05FJM 460087 IC50 = 18000 nM T35527 D05HOO 7244 IC50 > 100000 nM T35527 D06PRC 5281650 IC50 = 580 nM T35527 D07EAJ 10110469 IC50 > 50000 nM T35527 D07EGB 3610 IC50 > 10000 nM T35527 D07JRW 10179787 IC50 = 7900 nM T35527 D08WDW 10007601 Ki = 9000 nM T35527 D0B5GC 11349 IC50 > 100000 nM T35527 D0F1VR 44396194 IC50 = 47000 nM T35527 D0F9FG 46907602 IC50 = 3100 nM T35527 D0H8FG 637821 IC50 = 260 nM T35527 D0I6ZS 476857 IC50 = 3100 nM T35527 D0JL2T 5393152 IC50 > 100000 nM T35527 D0K0QU 11740143 IC50 = 280 nM T35527 D0M6KL 11211821 IC50 = 10700 nM T35527 D0MF5Y 5281614 IC50 = 950 nM T35527 D0NQ7I 10029508 IC50 = 50000 nM T35527 D0NU1W 636835 IC50 = 30000 nM T35527 D0P1LP 7090 IC50 = 100 nM T35527 D0Q0LD 15482063 Ki = 17000 nM T35527 D0U2YL 131820 IC50 = 640 nM T35527 D0US4S 5283159 IC50 = 15000 nM T35527 D0X4BT 425241 IC50 = 210 nM T35527 D0X4CI 9986835 IC50 = 700 nM T27889 D08EYQ 448281 IC50 = 0.44 nM T27889 CE1H5V 1382255 IC50 = 62000 nM T27889 C8P2UD 24827309 Ki = 7.5 nM T27889 CRS26D 24827437 Ki = 6.5 nM T27889 CD0ME8 24827440 Ki = 7 nM T27889 CG6WS4 24827547 Ki = 5.2 nM T27889 C0SEG1 24827658 Ki = 5.2 nM T27889 CUYB68 24827661 Ki = 6.6 nM T27889 CYP60C 24827781 Ki = 0.7 nM T27889 C79VFM 24827784 Ki = 920 nM T27889 C01XOT 24827913 Ki = 800 nM T27889 C9A0HU 24828308 Ki = 300 nM T27889 C5ESN2 24828309 Ki = 300 nM T27889 C7NS5H 24828310 Ki = 3000 nM T27889 CH8IC5 24828443 Ki > 10000 nM T27889 C02ZBM 24828444 Ki > 10000 nM T27889 CI0A7J 24828445 Ki = 8000 nM T27889 C7W5MA 24828578 Ki > 10000 nM T27889 C6FGD3 24828579 Ki > 10000 nM T27889 C98THQ 24828580 Ki > 10000 nM T27889 C74JBV 24829232 Ki > 10000 nM T27889 CP2LY7 25033280 Ki = 1.5 nM T27889 C4YKQ1 25033281 Ki = 7.1 nM T27889 CG75AN 44377126 Ki = 86 nM T27889 C06HJB 44446952 Ki = 1.5 nM T27889 CNK7X5 44446953 Ki = 90 nM T27889 CEB78N 44446954 Ki = 14 nM T27889 CMO78A 44446956 Ki = 1.5 nM T27889 CV6H2M 44446957 Ki = 1.3 nM T27889 CF4KE1 44446959 Ki = 2.2 nM T27889 CW9C0E 44446960 Ki = 2.4 nM T27889 CQB5M0 44446963 Ki = 37 nM T27889 C94POY 44446965 Ki = 2.2 nM T27889 CBX2U9 44446967 Ki = 0.9 nM T27889 CRZ6B3 44446968 Ki = 5.8 nM T27889 CY9O4I 44446969 Ki = 2.2 nM T27889 C4PQ7D 44446970 Ki = 6 nM T27889 C96KIY 44446972 Ki = 2.4 nM T27889 CK1EM5 44446974 Ki = 2.7 nM T27889 C4V6RZ 44446975 Ki = 2.5 nM T27889 CBL9E6 44446976 Ki = 2 nM T27889 CVYX54 44446979 Ki = 0.85 nM T27889 CAI9Z6 44446980 Ki = 35 nM T27889 C86KVP 44446984 Ki = 84 nM T27889 CXP2V4 44450296 Ki = 220 nM T27889 C29JUG 44450311 Ki = 0.4 nM T27889 C29YXI 44450312 Ki = 1.25 nM T27889 CC2IS3 44454957 Ki = 65 nM T27889 C1ESI2 44454959 Ki = 2.4 nM T27889 C8L0MV 44454960 Ki = 1.8 nM T27889 CBG6T0 44454987 Ki = 1.6 nM T27889 CN7UW3 44455013 Ki = 1.8 nM T27889 CC5L7S 44455015 Ki = 2300 nM T27889 C6KDT1 44455016 Ki = 1.4 nM T27889 CF4ML7 44455018 Ki = 6.9 nM T27889 CZI6S1 44455047 Ki = 320 nM T27889 C3UF6E 44455406 Ki = 860 nM T27889 CJG71N 44455407 Ki = 550 nM T27889 C0IR5W 44455428 Ki = 420 nM T27889 C62KSV 44455429 Ki = 84 nM T27889 CR9WL2 44455430 Ki = 1.4 nM T27889 CGH0S7 54589400 IC50 > 100000 nM T27889 D05JBC 98888 IC50 = 57000 nM T27889 D0N4RO 44377139 Ki = 1400 nM T27889 D0P0MP 24827312 Ki = 0.13 nM T55703 D08JAC 5288209 EC50 = 2372 nM T55703 CCV13B 307715 IC50 = 30000 nM T55703 CQIC85 1240497 IC50 > 30000 nM T55703 CHL2J7 2741694 IC50 = 130 nM T55703 C7H9EQ 4594798 IC50 > 30000 nM T55703 CAS81H 6437840 EC50 = 145 nM T55703 C8JOH2 6440160 EC50 = 245 nM T55703 CW1TB6 6505795 EC50 = 171 nM T55703 CT29IO 9339282 IC50 = 600 nM T55703 CX76JZ 11646381 EC50 = 154 nM T55703 C5E4NL 23847608 IC50 = 890 nM T55703 C6ZSN0 24099689 IC50 > 30000 nM T55703 C9Z6UG 25138295 IC50 = 0.155 nM T55703 CUY52L 53362669 EC50 = 1260 nM T55703 C5E0YI 53362728 EC50 = 954 nM T55703 CD6N5Z 72194831 IC50 = 4500 nM T55703 C9VKZ2 72194832 IC50 = 2500 nM T55703 C5I1UV 72194950 IC50 = 2200 nM T55703 CVRK75 72194951 IC50 = 360 nM T55703 CB24NZ 72194952 IC50 = 17 nM T55703 C2W1GC 72194954 IC50 = 160 nM T55703 CPX7Q3 72195086 IC50 > 10000 nM T55703 CCR0L6 72195223 IC50 = 350 nM T55703 C1WN6G 72195224 IC50 = 480 nM T55703 C3RPB9 72195225 IC50 = 3600 nM T55703 C46UJV 72195227 IC50 = 1100 nM T55703 CJ4IC1 72195368 IC50 = 920 nM T55703 CSXK92 72195505 IC50 = 830 nM T55703 C56OVE 72195508 IC50 = 76 nM T55703 CSI86X 72195642 IC50 = 270 nM T55703 CUB09N 72195775 IC50 = 17 nM T55703 CIA7P2 72195777 IC50 = 550 nM T55703 CF3JG8 72195779 IC50 = 120 nM T55703 C8PGY0 72195780 IC50 = 3 nM T55703 C6WE0U 72195781 IC50 = 120 nM T55703 C2R6BO 72195909 IC50 = 18 nM T55703 CYV4Z6 73890929 IC50 = 0.294 nM T55703 CWE0Z1 74983356 IC50 = 440 nM T55703 CFM87J 81689710 IC50 = 2.66 nM T55703 CW6ZH5 86272037 IC50 = 0.554 nM T55703 C3DMU6 86272278 IC50 = 2.65 nM T55703 CQA64O 86272279 IC50 > 3000 nM T55703 C5OLB6 86272531 IC50 = 140.6 nM T55703 CNT8M1 86297622 IC50 = 57.4 nM T55703 C5I8AV 86297623 IC50 = 3.9 nM T55703 C5C3FT 86303362 IC50 = 4.1 nM T55703 C8TMB0 86303363 IC50 = 4.5 nM T55703 C25JLT 86303514 IC50 = 6 nM T55703 CKM30G 86303515 IC50 = 3.4 nM T55703 CP7R0G 86303516 IC50 = 2.7 nM T55703 CKC43R 86303667 IC50 = 32.8 nM T55703 C7TO8Q 86303671 IC50 = 14.6 nM T55703 C42VEU 86303814 IC50 = 10 nM T55703 C9ES1B 86303815 IC50 = 6 nM T55703 C6A1DG 86304283 IC50 = 0.179 nM T55703 C0IZU4 86304284 IC50 = 170.3 nM T55703 C5JFM1 86304285 IC50 = 0.285 nM T55703 CKJI10 86304439 IC50 = 0.34 nM T55703 CGK31H 86304440 IC50 = 1.55 nM T55703 CJ7SI6 86304441 IC50 > 3000 nM T55703 C4CX7B 86304442 IC50 = 0.481 nM T55703 C9EMQ0 86304601 IC50 = 12.8 nM T55703 CK91QM 86304602 IC50 = 6.3 nM T55703 CV4Q5D 86304762 IC50 = 0.121 nM T55703 C4W7OE 90644283 IC50 = 3610 nM T55703 C1YW9K 90644284 IC50 = 60 nM T55703 C5LJG0 90644285 IC50 = 830 nM T55703 C6D7UF 117606941 IC50 = 9.61 nM T55703 C9NW1U 117606943 IC50 = 4.98 nM T55703 C8TI3G 117607480 IC50 = 5.47 nM T55703 CB0U6K 117607488 IC50 = 128 nM T55703 C9W1BQ 117607502 IC50 = 9.54 nM T55703 CC89FH 117607506 IC50 = 29.8 nM T55703 C40LSF 117607513 IC50 > 3000 nM T55703 CKI73Z 117607518 IC50 = 3.6 nM T55703 C0E1WB 117607520 IC50 = 10.8 nM T55703 CM78JQ 117607528 IC50 = 9.71 nM T55703 CAW25M 117607530 IC50 = 8.26 nM T55703 C07UOV 117607537 IC50 = 3.13 nM T55703 C95UFH 117607570 IC50 = 3.75 nM T55703 C3V1GL 117607574 IC50 = 6.28 nM T55703 CRJM60 117614486 IC50 = 53.3 nM T55703 CQ7S4B 117614487 IC50 = 14.1 nM T55703 CAKZ32 117614489 IC50 = 48.8 nM T55703 CGL3R6 117614609 IC50 = 0.235 nM T55703 C7KNV4 118053650 IC50 = 4.1 nM T55703 CBJ28X 118483320 IC50 = 5.73 nM T55703 C29OUV 118483422 IC50 = 4.88 nM T55703 C4E9LW 118483444 IC50 = 5.84 nM T55703 CFUQ68 118483473 IC50 = 9.06 nM T55703 C1G9YA 118674745 IC50 = 12.8 nM T55703 CS8AM9 118674749 IC50 = 90.1 nM T55703 CP9X4Y 118674754 IC50 = 381 nM T55703 CNCK26 118674756 IC50 = 20.8 nM T55703 C3YK2D 118674777 IC50 = 33.4 nM T55703 CR8W0P 118674778 IC50 = 171 nM T55703 CICJ02 118674788 IC50 = 153 nM T55703 CNZ14J 118674806 IC50 = 9.6 nM T55703 CG19QW 118722887 IC50 = 6.8 nM T55703 C8XHB1 118722888 IC50 = 5.31 nM T55703 CK1F3Y 118722889 IC50 = 3.94 nM T55703 C6E2GT 118722890 IC50 = 1470 nM T55703 C81YEC 118722891 IC50 > 3000 nM T55703 CI5WE1 118723219 IC50 > 3000 nM T55703 CBG74A 118723220 IC50 > 3000 nM T55703 C0C2ZD 118723221 IC50 > 3000 nM T55703 CTN6C4 118723222 IC50 = 8.38 nM T55703 CCN52L 118723223 IC50 = 1440 nM T55703 C1ZC8T 118723224 IC50 = 3760 nM T55703 CTN6R7 118723225 IC50 = 6.82 nM T55703 CJ29BC 118723226 IC50 = 5.26 nM T55703 CW4LE1 118723227 IC50 = 9.19 nM T55703 CC0V8J 118723228 IC50 = 0.829 nM T55703 CTXW94 118723229 IC50 = 1320 nM T55703 CODS97 118872290 IC50 = 4.55 nM T55703 C14DLY 118872292 IC50 = 5.14 nM T55703 C5IB6X 118872295 IC50 = 6.74 nM T55703 CN82DK 118872300 IC50 = 6.82 nM T55703 C94ZIC 118872302 IC50 = 6.99 nM T55703 CV4LB3 118872305 IC50 = 4.71 nM T55703 CP19ZK 118872306 IC50 = 7.53 nM T55703 C5PCN4 118872312 IC50 = 3.7 nM T55703 C4Q5DC 118872313 IC50 = 44.6 nM T55703 CK19OB 118872316 IC50 = 15.9 nM T55703 C61CQB 118872320 IC50 = 3.97 nM T55703 CX86IR 118872321 IC50 = 84.2 nM T55703 CZ32GQ 118872329 IC50 = 8.5 nM T55703 C6PT4Q 118872330 IC50 = 4.01 nM T55703 CJG56Z 118872333 IC50 = 6.36 nM T55703 C1Y4LH 118872342 IC50 = 6.42 nM T55703 CBQW26 118872343 IC50 = 3.71 nM T55703 CP47NS 118872352 IC50 = 4.12 nM T55703 CDI5O2 118872366 IC50 = 3.9 nM T55703 CWOX09 118872370 IC50 = 4.71 nM T55703 CE8RT5 122181975 IC50 = 3.3 nM T55703 CB3GT1 122181976 IC50 = 7.5 nM T55703 C5YD3R 122181977 IC50 = 4908 nM T55703 CD18WR 122181978 IC50 > 3000 nM T55703 C63NYG 122181979 IC50 = 83.2 nM T55703 CBE2G4 122181980 IC50 = 68.4 nM T55703 CNA61H 122181981 IC50 = 166 nM T55703 CTYV63 122181982 IC50 = 23 nM T55703 CPH0O2 122181983 IC50 = 29.3 nM T55703 C39LIA 122181984 IC50 = 196 nM T55703 C68UJQ 122181985 IC50 = 347 nM T55703 CDL2E5 122181986 IC50 = 137 nM T55703 CTZ2S6 122181987 IC50 = 821 nM T55703 CJK58R 122182099 IC50 = 719 nM T55703 CB8OX7 122182536 IC50 = 188 nM T55703 CRP96Y 122182537 IC50 = 9.7 nM T55703 C9Y1DW 122182538 IC50 = 89.5 nM T55703 CKC5B7 122182539 IC50 = 40.8 nM T18616 CYQ7L5 1365686 Ki = 292 nM T18616 CN8XM2 5311263 EC50 = 12 nM T18616 CLS96Y 6419701 EC50 = 67.61 nM T18616 COZF72 10322404 EC50 = 5.012 nM T18616 C7QRT8 11648176 EC50 = 0.83 nM T18616 C1F9GI 24882686 IC50 > 30000 nM T18616 CV86RF 44368508 EC50 = 8.128 nM T18616 C85ANH 46213949 IC50 > 8000 nM T18616 CET63X 46223906 EC50 = 6.3 nM T18616 CWF21Q 66552906 IC50 = 800 nM T18616 C57TYK 71569053 EC50 = 0.257 nM T18616 CSN3I7 71569056 EC50 = 1.81 nM T18616 CPT5S2 71718248 EC50 = 3 nM T18616 CKC4U7 71719457 EC50 = 6.1 nM T18616 C5P1CQ 71720690 EC50 = 3.388 nM T18616 D02LXI 10367662 IC50 > 30000 nM T18616 D0X0UR 5497152 EC50 = 140 nM T90935 C1Y7SN 13044112 IC50 = 2.5 nM T90935 CV57AQ 24768125 IC50 = 0.7 nM T90935 CJL02U 24801433 IC50 = 823 nM T90935 CL5M2P 145949885 IC50 = 203 nM T90935 CJ62VN 145950127 IC50 = 805 nM T90935 C38SNF 145951757 IC50 = 16900 nM T90935 CL2M9K 145951992 IC50 = 2.9 nM T90935 CP64UE 145952750 IC50 = 4.2 nM T90935 C06RXH 145955009 IC50 = 198 nM T90935 COG1C8 145957811 IC50 = 6.3 nM T90935 C4EX5L 145959286 IC50 = 0.1 nM T90935 C9KNH4 145959543 IC50 = 3.3 nM T90935 C4EXJ0 145959627 IC50 = 5.5 nM T08647 D0E3TC 44259 IC50 = 11.8 nM T08647 CV63UL 67240318 IC50 > 5000 nM T08647 C9WGB8 127035904 IC50 = 3500 nM T08647 C2AN7T 134611886 IC50 > 100000 nM T08647 D0X8BU 71718651 IC50 = 1500 nM T41371 D0K0SB 5487121 IC50 = 0.01 ug.mL-1 T41371 C5V7WC 443301 IC50 = 730000 nM T41371 CURX40 505897 IC50 = 0.027 ug.mL-1 T41371 CPW64U 513190 IC50 = 0.0065 ug.mL-1 T41371 C01FLO 513191 IC50 = 0.24 ug.mL-1 T41371 CDO7V0 513195 IC50 > 2.5 ug.mL-1 T41371 CBC2X6 513514 IC50 = 0.18 ug.mL-1 T41371 CUF0O8 513515 IC50 = 0.28 ug.mL-1 T41371 CPY7E6 513516 IC50 > 2.5 ug.mL-1 T41371 C4S1FK 513517 IC50 = 0.42 ug.mL-1 T41371 CA2DH4 513518 IC50 = 0.03 ug.mL-1 T41371 CGHZ21 513519 IC50 = 0.03 ug.mL-1 T41371 C6O3KY 513521 IC50 = 0.14 ug.mL-1 T41371 CA2PT8 513522 IC50 = 0.07 ug.mL-1 T41371 CPFZ49 513523 IC50 = 0.09 ug.mL-1 T41371 C1D6JS 513524 IC50 = 0.6 ug.mL-1 T41371 CFW87P 513525 IC50 = 0.17 ug.mL-1 T41371 C1ZUA5 513526 IC50 = 0.26 ug.mL-1 T41371 C8VG7Q 513527 IC50 = 0.39 ug.mL-1 T41371 C9Z8DC 513528 IC50 > 2.5 ug.mL-1 T41371 CY12DB 513529 IC50 = 0.021 ug.mL-1 T41371 CS6Z3K 513530 IC50 = 0.034 ug.mL-1 T41371 CC0MO4 513531 IC50 = 0.032 ug.mL-1 T41371 CYN70W 513532 IC50 = 0.019 ug.mL-1 T41371 CL69FN 513533 IC50 = 0.04 ug.mL-1 T41371 CID52Q 513534 IC50 = 0.025 ug.mL-1 T41371 CX0DF4 513535 IC50 = 0.022 ug.mL-1 T41371 C7OVP1 513536 IC50 = 0.028 ug.mL-1 T41371 CI63EA 513537 IC50 = 0.02 ug.mL-1 T41371 CMU52E 513538 IC50 = 0.02 ug.mL-1 T41371 C9WJ7A 513539 IC50 = 0.019 ug.mL-1 T41371 CYIR84 513540 IC50 = 0.06 ug.mL-1 T41371 CX8U6J 513541 IC50 = 0.13 ug.mL-1 T41371 C1IWR7 513542 IC50 = 0.11 ug.mL-1 T41371 CM2PA9 513543 IC50 = 0.013 ug.mL-1 T41371 CA41EO 513544 IC50 = 0.12 ug.mL-1 T41371 C07FSE 513545 IC50 = 0.5 ug.mL-1 T41371 CJ63FU 513546 IC50 = 1.2 ug.mL-1 T41371 C2AE5N 513547 IC50 = 0.2 ug.mL-1 T41371 CO3P1B 513548 IC50 = 0.28 ug.mL-1 T41371 C03COZ 513549 IC50 = 0.7 ug.mL-1 T41371 CCK01G 513550 IC50 = 0.42 ug.mL-1 T41371 CFC89S 513551 IC50 = 0.2 ug.mL-1 T41371 CYD59Z 513553 IC50 = 0.11 ug.mL-1 T41371 CSW1L6 513554 IC50 = 0.28 ug.mL-1 T41371 CR6U4F 513555 IC50 = 0.077 ug.mL-1 T41371 C7V1HP 513556 IC50 = 0.36 ug.mL-1 T41371 CU7EN4 513557 IC50 > 2.5 ug.mL-1 T41371 C3MGB1 513558 IC50 = 0.0076 ug.mL-1 T41371 C8NJH5 513559 IC50 = 0.013 ug.mL-1 T41371 CB2HR7 513560 IC50 = 0.06 ug.mL-1 T41371 CXY19L 513561 IC50 = 0.054 ug.mL-1 T41371 C86GVN 513562 IC50 = 0.02 ug.mL-1 T41371 CWO14D 513563 IC50 = 0.031 ug.mL-1 T41371 C4BK6G 513564 IC50 = 0.12 ug.mL-1 T41371 C62INT 513565 IC50 = 0.16 ug.mL-1 T41371 C5ZE7A 513567 IC50 = 0.031 ug.mL-1 T41371 CK2F3C 513568 IC50 = 0.037 ug.mL-1 T41371 CF6S3J 513569 IC50 = 0.023 ug.mL-1 T41371 CD6YV2 513570 IC50 = 0.01 ug.mL-1 T41371 C6YJZ3 513571 IC50 = 0.037 ug.mL-1 T41371 CQ4VK8 513572 IC50 = 0.013 ug.mL-1 T41371 C14KHS 513573 IC50 = 0.015 ug.mL-1 T41371 CU7TN2 513574 IC50 = 0.009 ug.mL-1 T41371 CNM2E6 513575 IC50 = 0.018 ug.mL-1 T41371 C2CIF6 513576 IC50 = 0.02 ug.mL-1 T41371 CSV3K1 513578 IC50 = 0.018 ug.mL-1 T41371 C0QU4S 3006554 IC50 = 0.3 ug.mL-1 T41371 C3SYJ6 3006557 IC50 = 0.7 ug.mL-1 T41371 C4ADJ0 3006558 IC50 = 1.9 ug.mL-1 T41371 C1CWK7 3006559 IC50 > 2.5 ug.mL-1 T41371 CLE8Q0 3006602 IC50 = 0.13 ug.mL-1 T41371 C41RKF 3006607 IC50 = 0.03 ug.mL-1 T41371 CAJW83 5495616 IC50 = 0.01 ug.mL-1 T41371 C7F5GR 5496295 IC50 = 0.027 ug.mL-1 T41371 CRPS35 5496296 IC50 = 0.015 ug.mL-1 T41371 CP47ZY 9897006 IC50 = 2.2 ug.mL-1 T41371 CJG0F4 9950619 IC50 = 90000 nM T41371 CJ8D3I 9992643 IC50 = 195000 nM T41371 C53KWH 10001147 IC50 = 30000 nM T41371 C69TOZ 10040630 IC50 = 185000 nM T41371 C5KXD0 10065189 IC50 > 900000 nM T41371 CTE5V1 10387239 IC50 = 25000 nM T41371 CD9GF0 11722365 IC50 = 140000 nM T41371 C1UB4S 12443047 IC50 > 900000 nM T41371 CTZ7U3 44273197 IC50 = 50000 nM T41371 CT73SP 44299515 IC50 > 900000 nM T41371 C8NK6B 44299557 IC50 = 290000 nM T41371 C6OKU8 44299559 IC50 > 900000 nM T41371 CT26ZR 44299601 IC50 > 900000 nM T41371 CPD72Y 44299623 IC50 > 900000 nM T41371 CTD14E 44299624 IC50 > 900000 nM T41371 CZH90M 44299667 IC50 > 900000 nM T41371 CR35XC 44299679 IC50 = 200000 nM T41371 C9ASB8 44299688 IC50 = 480000 nM T41371 CKR8C0 44299690 IC50 = 600000 nM T41371 C9BT2I 44299734 IC50 = 300000 nM T41371 C4MYW7 44299739 IC50 > 900000 nM T41371 CI80LE 44299741 IC50 = 400000 nM T41371 CZ0SN1 44327812 IC50 = 0.04 ug.mL-1 T41371 CT0RD6 44327813 IC50 = 0.18 ug.mL-1 T41371 CBD02P 44327815 IC50 = 0.105 ug.mL-1 T41371 CW62ES 44327844 IC50 = 0.04 ug.mL-1 T41371 CEBU87 44328154 IC50 = 0.17 ug.mL-1 T41371 C4VT5B 44328158 IC50 = 1 ug.mL-1 T41371 CF32XM 44328159 IC50 = 0.6 ug.mL-1 T41371 CP1M9A 44328236 IC50 = 0.64 ug.mL-1 T41371 CB8N4J 44328264 IC50 = 0.43 ug.mL-1 T41371 CRN1U0 44328265 IC50 = 2.4 ug.mL-1 T41371 CE7Y6W 44328266 IC50 = 4.5 ug.mL-1 T41371 C4ZWG5 44328287 IC50 = 0.19 ug.mL-1 T41371 C4JP3K 44328288 IC50 = 0.045 ug.mL-1 T41371 CL9B4J 44328323 IC50 = 0.2 ug.mL-1 T41371 C89WVO 44328324 IC50 = 0.13 ug.mL-1 T41371 C6Z0GF 44328325 IC50 = 15 ug.mL-1 T41371 C4KFJ5 44328366 IC50 > 2.5 ug.mL-1 T41371 CJ46ES 44328367 IC50 = 1.4 ug.mL-1 T41371 CN57VK 44328373 IC50 = 30 ug.mL-1 T41371 CWV13J 44328377 IC50 = 0.5 ug.mL-1 T41371 CAZI30 44328453 IC50 = 0.05 ug.mL-1 T41371 CB4WT0 44328489 IC50 = 0.024 ug.mL-1 T41371 CC9B5S 44328506 IC50 = 8 ug.mL-1 T41371 CQ7OU3 44328546 IC50 = 0.043 ug.mL-1 T41371 C27BEG 44328632 IC50 = 0.15 ug.mL-1 T41371 CZ4CI2 44328674 IC50 = 0.055 ug.mL-1 T41371 CI6HE4 44328726 IC50 = 0.04 ug.mL-1 T41371 CV6P3O 44366372 IC50 = 5000 nM T41371 C0PS3L 44366495 IC50 > 1000000 nM T41371 C4VZH0 44366502 IC50 = 150000 nM T41371 CT4WR7 44366508 IC50 > 1000000 nM T41371 CR5F6V 44366512 IC50 > 1000000 nM T41371 CWHL79 44366631 IC50 > 1000000 nM T41371 C9EVH8 44366643 IC50 = 45000 nM T41371 CJP9I8 44366648 IC50 > 1000000 nM T41371 CXLF25 44366668 IC50 = 130000 nM T41371 C6L3ZF 44366683 IC50 = 180000 nM T41371 C3W5JQ 44366684 IC50 = 140000 nM T41371 D0Y0KV 3013049 IC50 = 0.55 ug.mL-1 T69085 D08JIS 46926788 IC50 = 7500 nM T69085 D01OLO 9820526 IC50 = 8 nM T69085 D02LCL 23626877 IC50 = 10000 nM T69085 CBW19J 181498 IC50 = 1500 nM T69085 C08KAG 441796 IC50 = 40 nM T69085 C4VG9X 9863590 IC50 = 20 nM T69085 CQ7J0C 9907138 IC50 > 3000 nM T69085 C2TS1U 9907182 IC50 = 3 nM T69085 C6DBO0 9910975 IC50 = 50 nM T69085 CLWO04 10065309 IC50 = 100 nM T69085 C64YXB 10067871 IC50 = 45 nM T69085 CUE3O7 10245314 IC50 = 35 nM T69085 C7J2GH 10336479 IC50 = 100000 nM T69085 C10MCP 10407641 IC50 = 20 nM T69085 CD0M8B 10499355 IC50 = 4000 nM T69085 CN0MX6 10525196 IC50 > 10000 nM T69085 C48SVD 10552343 IC50 > 10000 nM T69085 CKC1V4 10574522 IC50 > 10000 nM T69085 C9EUI1 10574991 IC50 = 10000 nM T69085 CN9S4F 10622840 IC50 > 10000 nM T69085 CT0QH3 10624842 IC50 = 600 nM T69085 CQ8W9A 10666813 IC50 = 300 nM T69085 C2GY5Z 10666814 IC50 = 1700 nM T69085 CJ16AD 10716177 IC50 > 10000 nM T69085 CJ5NW8 10716536 IC50 > 10000 nM T69085 C6C0JV 10716588 IC50 = 500 nM T69085 COE42S 10717756 IC50 > 30000 nM T69085 CNT0E3 10740841 IC50 = 100 nM T69085 C3XI4G 10741644 IC50 > 10000 nM T69085 C61PDW 10741998 IC50 = 400 nM T69085 C7K2EB 10763720 IC50 = 200 nM T69085 CON93J 10764421 IC50 > 10000 nM T69085 CB40RO 10786213 IC50 > 10000 nM T69085 C7BAM8 10787015 IC50 = 300 nM T69085 CGRH71 10811870 IC50 > 10000 nM T69085 C3GRB1 10813496 IC50 = 8000 nM T69085 CJ9OH7 11538129 IC50 = 10000 nM T69085 CVS32L 11560956 IC50 = 1938 nM T69085 CN5R7T 11696956 IC50 = 5000 nM T69085 CW04NP 11842418 IC50 = 5500 nM T69085 CBC08P 11846124 EC50 = 318 nM T69085 C0C5AZ 16129582 IC50 = 704 nM T69085 CK7JE6 16752764 IC50 = 5000 nM T69085 C1JG8L 25017847 IC50 = 10000 nM T69085 C6O4MS 25017848 IC50 = 3300 nM T69085 CMAH54 25017849 IC50 = 500 nM T69085 CSYN01 42631933 IC50 = 5500 nM T69085 CX3AJ7 42632173 IC50 = 1200 nM T69085 CBQ0A6 44202126 IC50 = 30000 nM T69085 CKD03R 44241655 IC50 = 100 nM T69085 CA8DQ9 44289488 IC50 = 1000 nM T69085 C5T9MD 44320262 IC50 = 400 nM T69085 CA78EB 44320323 IC50 = 300 nM T69085 CP3RW2 44320513 IC50 = 98 nM T69085 C3G4YN 44320524 IC50 = 2000 nM T69085 CRWI45 44320559 IC50 = 210 nM T69085 CO3P4J 44320570 IC50 = 4400 nM T69085 CAX8F5 44440161 IC50 = 3700 nM T69085 CK9H1G 44440214 IC50 = 8091 nM T69085 CDF70Q 44440215 IC50 = 7723 nM T69085 CK8L4U 44440216 IC50 > 10000 nM T69085 CM2E3N 44440217 IC50 = 19331 nM T69085 CWL30H 44440218 IC50 = 29891 nM T69085 C6RD3G 44440219 IC50 = 6268 nM T69085 CIAJ70 44440220 IC50 = 4272 nM T69085 C52CDB 44440221 IC50 = 6995 nM T69085 C2OC7L 44440222 IC50 = 14667 nM T69085 CFZS24 44440223 IC50 = 3883 nM T69085 CSA87R 44440224 IC50 = 2807 nM T69085 CH76CV 44440225 IC50 = 1769 nM T69085 CP80UK 44440226 IC50 = 741 nM T69085 CFI06W 44440227 IC50 = 2770 nM T69085 CKSO82 44440228 IC50 = 2028 nM T69085 C8HWI1 44440229 IC50 = 2497 nM T69085 CVD97U 44440230 IC50 = 813 nM T69085 C1B0TO 44440234 IC50 = 807 nM T69085 CS5PY4 44440235 IC50 = 21160 nM T69085 C9AV4C 44440236 IC50 = 3845 nM T69085 CJVG30 44443369 IC50 > 300 nM T69085 CS5E1A 44443376 IC50 > 1000 nM T69085 CI94CU 44443382 IC50 > 3000 nM T69085 C9WL4G 44443383 IC50 > 3000 nM T69085 CZV7S2 44443402 IC50 > 300 nM T69085 CW9O2X 45267090 IC50 = 71 nM T69085 CF7MG2 46932984 IC50 = 5700 nM T69085 C2Z1HP 46933276 IC50 = 14000 nM T69085 C6AN4W 46933278 IC50 > 500000 nM T69085 CLV8G5 46933420 IC50 = 4300 nM T69085 C1HI2W 51346940 IC50 = 100 nM T69085 C5GPU9 51346941 IC50 = 310 nM T69085 CI5FZ2 53363123 EC50 = 130 nM T69085 C9JTA1 53493058 IC50 = 5200 nM T69085 CH4B5I 53493059 IC50 = 6000 nM T69085 CCG3H2 54580285 IC50 = 160 nM T69085 CHN37L 54581281 IC50 = 4000 nM T69085 CB4TJ8 54581287 IC50 = 120 nM T69085 CT3JS6 54581291 IC50 = 3000 nM T69085 CM7H3P 54581292 IC50 = 40 nM T69085 C6B2UL 54582304 IC50 = 620 nM T69085 C1FR4Q 54582305 IC50 = 130 nM T69085 CP4HV1 54582306 IC50 = 40 nM T69085 CFG68S 54582307 IC50 = 50 nM T69085 C1OM6E 54583278 IC50 = 200 nM T69085 CNE41S 54583279 IC50 = 5100 nM T69085 CMCL04 54583281 IC50 = 630 nM T69085 CTQ70F 54583282 IC50 = 930 nM T69085 CM1TU0 54584242 IC50 = 250 nM T69085 CP6K3I 54584243 IC50 = 1400 nM T69085 CR4E7O 54584244 IC50 = 500 nM T69085 CT16HO 54585212 IC50 = 20 nM T69085 CI8ZH6 54587176 IC50 = 40 nM T69085 C1V8HM 54587177 IC50 = 290 nM T69085 CO1JB2 54587178 IC50 = 330 nM T69085 C3JAW8 54587179 IC50 = 3000 nM T69085 CGC25V 57620293 IC50 = 11900 nM T69085 CUCW84 76324956 IC50 = 1600 nM T69085 CK2HX0 76335838 IC50 = 1300 nM T69085 C9QD8T 90668286 IC50 = 5400 nM T69085 C3F4LZ 90668287 IC50 = 64000 nM T69085 CI9R8V 101135598 IC50 = 29000 nM T69085 CW5AC6 118716125 IC50 = 500 nM T69085 CK4VQ0 118716126 IC50 > 10000 nM T69085 C48PKT 118716127 IC50 > 10000 nM T69085 CH1OL7 118716128 IC50 = 10000 nM T69085 CQ45JC 118716129 IC50 = 9400 nM T69085 CQ6G7M 118716130 IC50 = 9400 nM T69085 CPY16H 118716131 IC50 = 6100 nM T69085 C0UA6E 118716132 IC50 = 8500 nM T69085 CVRK59 118716133 IC50 = 10000 nM T69085 CVZ56P 118716134 IC50 = 1900 nM T69085 C5P0LJ 118716135 IC50 = 830 nM T69085 CB1AL4 118716136 IC50 = 760 nM T69085 C6JZF4 118716171 IC50 = 69600 nM T69085 C7X4TL 155563713 IC50 = 7000 nM T69085 D04HFC 44443385 IC50 = 68 nM T69085 D05PTT 5281792 IC50 = 16200 nM T69085 D0C1UM 161749 IC50 = 65 nM T69085 D0T1XE 264751 IC50 = 110 nM T69085 D0Y9AQ 402628 IC50 = 1067 nM T67754 C6KL0E 120267 EC50 = 2710 nM T67754 C6PJH5 1281059 IC50 = 3900 nM T67754 CSLC42 10539503 EC50 = 1200 nM T67754 CGUL70 11161014 EC50 = 1600 nM T67754 C98SFK 11215125 EC50 = 12 nM T67754 C3KV8G 11337049 EC50 = 56 nM T67754 CEC1I0 11570071 EC50 = 479 nM T67754 CJZI83 11650037 EC50 = 32 nM T67754 CJG04D 11652143 EC50 = 110 nM T67754 C02PRC 11652144 EC50 = 110 nM T67754 CI45SU 11708995 EC50 = 9541 nM T67754 CE8Y2K 11708996 EC50 = 9500 nM T67754 CU87IH 11709421 EC50 = 28 nM T67754 CMQ53X 11717063 EC50 = 470 nM T67754 CMZ8A9 11738113 EC50 = 18 nM T67754 C8Y9UE 25022659 EC50 = 160 nM T67754 C76OAY 25033279 EC50 = 1100 nM T67754 CZVD61 44445993 EC50 = 101870 nM T67754 C5YT8Q 44445994 EC50 = 8 nM T67754 CH6JG2 44445995 EC50 = 9 nM T67754 C1CWL3 44445996 EC50 = 9 nM T67754 COCN04 44445997 EC50 = 8 nM T67754 CH7B6P 44445998 EC50 = 28 nM T67754 CHC7B2 44445999 EC50 = 15 nM T67754 CT3K7A 44446000 EC50 = 116 nM T67754 CX4GL3 44446001 EC50 = 6000 nM T67754 CP8YB2 44446002 EC50 = 13 nM T67754 C9SAU2 44446003 EC50 = 52 nM T67754 CM8QY1 44453155 EC50 = 38000 nM T67754 C5UA3Y 44453190 EC50 = 24000 nM T67754 C6FT4W 44453258 EC50 = 8.3 nM T67754 CK4Y2Z 44453284 EC50 = 8.7 nM T67754 C8OI7M 44453313 EC50 = 360 nM T67754 C05CIM 44453349 EC50 = 1000 nM T67754 C9Y3LT 44453389 EC50 = 21 nM T67754 CF7CW3 44453393 EC50 = 1300 nM T67754 CUI82D 44453394 EC50 = 800 nM T67754 C2KO4M 44453424 EC50 = 840 nM T67754 CXEY56 44453425 EC50 = 25000 nM T67754 CRG04U 44453426 EC50 = 2200 nM T67754 C5XWH9 44453427 EC50 = 490 nM T67754 CE84NS 44453451 EC50 = 570 nM T67754 CQ8YT3 44453456 EC50 = 2300 nM T67754 CY1J7L 44453548 EC50 = 30 nM T67754 C94OXY 44453549 EC50 = 2000 nM T67754 C8FO7G 44453550 EC50 = 950 nM T67754 CJ3C2R 44453551 EC50 = 4.7 nM T67754 CC8HF2 44453553 EC50 = 300 nM T67754 C2LTU9 44453554 EC50 = 50 nM T67754 CYV0F1 44453632 EC50 = 3100 nM T67754 C5HYT0 44455082 EC50 = 3240 nM T67754 C18PVX 44455257 EC50 = 4700 nM T67754 CBNX36 44455282 EC50 = 17000 nM T67754 CRID29 44455318 EC50 = 6300 nM T67754 CY7R4T 44455319 EC50 = 8500 nM T67754 CFK1E8 44455350 EC50 > 10000 nM T67754 CC94PQ 44455383 EC50 = 660 nM T67754 CL3CP4 44455384 EC50 = 25000 nM T67754 C8K2WT 44455385 EC50 = 2600 nM T67754 CFO8A7 44455403 EC50 = 52000 nM T29678 D03FLC 3878 IC50 = 10000 nM T29678 D08HQK 5411 IC50 = 490 nM T29678 D0C7ET 11174599 IC50 = 14 nM T29678 D0E4DW 1775 Ki = 53370 nM T29678 D0H0KB 5070 IC50 = 2200 nM T29678 D0X0RI 4178 IC50 = 2900 nM T29678 D0Y5UG 2160 IC50 = 3100 nM T29678 D00BUR 216327 IC50 > 1000 nM T29678 D04JZH 11659955 IC50 = 12800 nM T29678 D04PER 49836093 IC50 = 600 nM T29678 D0K9IF 71666749 IC50 > 30000 nM T29678 D0O7QA 46840946 IC50 = 110 nM T29678 D0OX9F 16046068 IC50 = 13000 nM T29678 D0P5CM 56945146 IC50 > 33000 nM T29678 D0D1GV 9907241 IC50 = 1310 nM T29678 D0EC2K 60803 IC50 = 2550 nM T29678 CBK0G3 101313 Ki = 133560 nM T29678 C4OA7P 101314 Ki = 65560 nM T29678 C9LY7B 246391 Ki = 78420 nM T29678 C6D1LY 246499 Ki = 50400 nM T29678 CAG8Z4 269700 Ki = 337800 nM T29678 CFBM96 296732 IC50 = 40600 nM T29678 CJ8S9I 347569 Ki = 21800 nM T29678 C2T0DL 619974 Ki = 108070 nM T29678 CRK79S 787185 Ki = 20300 nM T29678 CPN25U 998021 IC50 = 240 nM T29678 C9L1HS 3586494 Ki = 16010 nM T29678 CB7H0W 5179365 Ki = 18270 nM T29678 C9ZT3K 9799052 IC50 = 820 nM T29678 CY30OZ 9819588 IC50 = 1140 nM T29678 CREZ06 9928808 IC50 = 4160 nM T29678 CMNO90 9974422 IC50 = 2200 nM T29678 C71ZGK 10316911 IC50 = 630 nM T29678 CR04QX 11032700 IC50 > 25000 nM T29678 CKB2G6 11780499 IC50 = 3870 nM T29678 CH8K2V 11780892 IC50 = 8810 nM T29678 C78UQR 11818545 IC50 = 2700 nM T29678 CRS3M1 13590017 IC50 = 1400 nM T29678 CHW13G 16040159 IC50 = 1500 nM T29678 CPCZ62 16040329 IC50 = 2800 nM T29678 C01EDT 16723427 IC50 = 17900 nM T29678 C8XUJ2 16725022 IC50 = 10100 nM T29678 C7C5OQ 18673182 IC50 = 21400 nM T29678 CL73HJ 21589240 IC50 = 0.0061 nM T29678 C5V2PF 22149197 IC50 = 3230 nM T29678 CAL57W 22149198 IC50 = 1390 nM T29678 CNM8X9 22149200 IC50 = 6030 nM T29678 C13HDG 22149207 IC50 = 2670 nM T29678 CYU64Q 22149216 IC50 = 1970 nM T29678 CUI6D7 22149230 IC50 = 2380 nM T29678 CNT32Z 22149267 IC50 = 4310 nM T29678 CH76LZ 22149271 IC50 = 1200 nM T29678 C2LUF7 22149278 IC50 = 3250 nM T29678 CG9S2U 22149289 IC50 = 9450 nM T29678 CL14RW 22149294 IC50 = 760 nM T29678 CGBU69 22149297 IC50 = 860 nM T29678 CCU53Q 22149327 IC50 > 25000 nM T29678 CMRN02 22149337 IC50 = 3900 nM T29678 CCY65J 22149344 IC50 = 2110 nM T29678 C6X0LN 22149356 IC50 = 4300 nM T29678 CFYW59 22149360 IC50 = 5030 nM T29678 CPXW92 22149373 IC50 = 1480 nM T29678 CJ25GQ 22371496 IC50 > 100000 nM T29678 CF75YB 24857856 IC50 = 100 nM T29678 CWF5Z3 25143506 IC50 > 30000 nM T29678 CP72MB 25159060 IC50 = 10000 nM T29678 C62NRA 44337110 IC50 = 1760 nM T29678 C4K5MJ 44337198 IC50 = 7110 nM T29678 CNB2Q7 44337215 IC50 = 5440 nM T29678 CP92BO 44337462 IC50 = 3350 nM T29678 CSMF57 44337512 IC50 = 4950 nM T29678 C85VGK 44337552 IC50 = 13750 nM T29678 C01UWF 44540282 IC50 > 33000 nM T29678 CN64WQ 44544347 IC50 = 8100 nM T29678 CEQ60V 44574939 IC50 = 1400 nM T29678 C31EXK 44574990 IC50 = 2500 nM T29678 C5YCD0 44574991 IC50 = 200 nM T29678 CER76K 44585595 IC50 = 350 nM T29678 C40BIM 45139151 IC50 = 429 nM T29678 CS5EJ1 46841648 IC50 = 2044 nM T29678 CRE97F 46841787 IC50 = 398 nM T29678 CBXW47 50899559 IC50 = 70 nM T29678 C06OXV 52920492 IC50 = 29000 nM T29678 C47GJP 52941142 IC50 = 360 nM T29678 C31XZV 52942252 IC50 = 18000 nM T29678 C4VE8S 52942340 IC50 = 1000 nM T29678 C3K0RO 52943146 IC50 = 8200 nM T29678 C9QAL2 52943533 IC50 = 1600 nM T29678 CH54UW 52944738 IC50 = 470 nM T29678 CU5CL0 52945245 IC50 = 5000 nM T29678 CDN9Y8 52945882 IC50 = 120 nM T29678 CI5BU7 52945890 IC50 = 670 nM T29678 CM2W7J 52945969 IC50 = 2200 nM T29678 CEK18S 52947191 IC50 = 1200 nM T29678 CJ6OG2 52947194 IC50 = 9100 nM T29678 C4X3KP 52947201 IC50 = 1000 nM T29678 CAQ8V0 52947207 IC50 = 1000 nM T29678 C0NZ9X 52948309 IC50 = 50 nM T29678 C6B0LV 52949221 IC50 = 1000 nM T29678 CJFG89 52949235 IC50 = 6200 nM T29678 CBC8U2 52949503 IC50 = 1600 nM T29678 C1LBT3 52949586 IC50 = 3900 nM T29678 CMS2F7 53239561 IC50 = 65000 nM T29678 CXEH21 56595883 IC50 = 4200 nM T29678 CGUA26 57331668 IC50 > 30000 nM T29678 C4FH0W 58118983 IC50 = 400 nM T29678 CM1G2P 59568656 IC50 > 30000 nM T29678 CA7NI3 60201088 IC50 > 33000 nM T29678 C1YQ8J 60201256 IC50 > 33000 nM T29678 CC82DM 65459349 IC50 = 16000 nM T29678 CT1YQ7 68680505 IC50 = 6900 nM T29678 CBH6T3 69003776 IC50 > 33000 nM T29678 C2MC6B 71522734 IC50 = 0.2 nM T29678 CM1B0W 71523649 IC50 = 17000 nM T29678 C0AO1Y 71556159 IC50 = 29 nM T29678 CJXK67 71559365 IC50 = 4.2 nM T29678 C9MUK3 71716856 IC50 = 149 nM T29678 CUG2V3 71716866 IC50 = 276 nM T29678 CX4IG6 72164684 IC50 = 1500 nM T29678 CM9KD6 76309675 Ki = 61070 nM T29678 C15BSO 86270136 IC50 = 14 nM T29678 CTG76E 86687532 IC50 = 2100 nM T29678 C1BIF8 90026208 IC50 = 2 nM T29678 C26BZK 91666633 IC50 = 7 nM T29678 C7NLE8 91809347 IC50 = 20 nM T29678 CNFW42 117608566 IC50 = 10 nM T29678 CC5N9I 117737142 IC50 = 2200 nM T29678 C9KV7L 117993993 IC50 = 9800 nM T29678 C7HJ6B 118126600 IC50 = 3500 nM T29678 C7AYV5 118540795 IC50 = 2.519 nM T29678 CR8TX9 118708662 IC50 = 41 nM T29678 C9JL4Y 118937760 IC50 = 4000 nM T29678 C9K5RV 122513516 IC50 > 20000 nM T29678 C09QIY 127047645 IC50 = 2600 nM T29678 CZ5H2B 132020452 IC50 = 16000 nM T29678 C9WC1S 135440609 IC50 > 24000 nM T29678 CWLX83 135443502 IC50 = 10090 nM T29678 CZ6WT3 135469086 IC50 = 1950 nM T29678 C9Q8GD 135568476 IC50 = 3290 nM T29678 CMC7Q6 135568488 IC50 = 4360 nM T29678 CN7J9F 135568497 IC50 > 25000 nM T29678 C3YB0A 135568523 IC50 = 1920 nM T29678 CL43OY 135568535 IC50 = 2020 nM T29678 CL04YV 137637468 IC50 = 0.28 nM T29678 CQN5I0 137637863 EC50 = 5.3 nM T29678 C5B1PR 137639568 EC50 = 120 nM T29678 C5I4EF 137648593 EC50 = 79 nM T29678 CK7PN3 145969142 IC50 = 1500 nM T29678 CZN0U6 145982478 IC50 = 2760 nM T29678 C8Q2EG 145988110 IC50 = 920 nM T29678 COZ54G 155523716 IC50 = 1600 nM T29678 CE3H4Z 155567528 IC50 = 120 nM T29678 D01AGR 24857857 IC50 = 1100 nM T29678 D02CQN 52945923 IC50 = 110 nM T29678 D06GQO 10955473 IC50 = 17350 nM T29678 D07FEO 190902 IC50 = 2030 nM T29678 D0FF6S 16038374 IC50 = 7180 nM T29678 D0O0JO 52948346 IC50 = 1200 nM T29678 D0O2RN 22149251 IC50 = 2660 nM T29678 D0P8TL 56947150 IC50 = 1 nM T29678 D0W2BP 46032908 IC50 = 1900 nM T30085 D01TNW 9887712 IC50 = 0.49 nM T30085 D04DXA 46908929 IC50 = 2.9 nM T30085 D06ALD 11949646 EC50 = 3 nM T30085 D08DFX 24812758 IC50 = 2.2 nM T30085 D0Q3VE 44814423 IC50 = 0.877 nM T30085 D07FBM 10453870 IC50 = 7.38 nM T30085 D0IJ0U 11988953 IC50 = 2.26 nM T30085 D0OR3G 25195624 IC50 = 5600 nM T30085 D0U7IL 24831714 IC50 = 1.5 nM T30085 C5ZBT0 646189 EC50 = 31100 nM T30085 CG1YL3 649241 EC50 > 50000 nM T30085 CM8QN1 658293 EC50 = 4600 nM T30085 CBA5C7 658756 EC50 = 11000 nM T30085 C54XQN 658758 EC50 = 34700 nM T30085 CI1DB0 780938 EC50 > 50000 nM T30085 CQB7O9 990391 EC50 = 8980 nM T30085 C7BS0Y 1226045 IC50 = 14700 nM T30085 C6D3EB 2822337 IC50 = 1400 nM T30085 CC39KX 2868088 EC50 = 40400 nM T30085 C32ZMW 2868153 EC50 = 19100 nM T30085 COCX40 2868345 EC50 = 3850 nM T30085 C5C7QP 2868397 EC50 = 16200 nM T30085 C59HJS 2868621 EC50 > 50000 nM T30085 CNG6Q5 2895998 EC50 = 5920 nM T30085 CXWS61 3086055 IC50 = 18700 nM T30085 C1R8VD 6474295 IC50 = 33300 nM T30085 CZI0R5 6918439 Ki = 4 nM T30085 CAP56Y 9797582 EC50 = 290 nM T30085 C1U6RK 9798876 EC50 = 5 nM T30085 CIX6M9 9800802 IC50 = 1 nM T30085 CD1H4F 9819601 EC50 = 540 nM T30085 C17EZH 9839914 EC50 = 623 nM T30085 C2HYT9 9841810 EC50 = 8 nM T30085 CP13LD 9842444 EC50 = 1200 nM T30085 CF9B2C 9862956 EC50 = 22 nM T30085 C9WKF7 9863600 EC50 = 480 nM T30085 C2FSB0 9863601 EC50 > 2 nM T30085 CV8U4S 9864271 EC50 = 630 nM T30085 C0SL7N 9883971 EC50 = 1200 nM T30085 CXW9J8 9886174 IC50 = 22 nM T30085 CTZ61Y 9906141 EC50 = 710 nM T30085 CNQ04U 9928743 EC50 = 430 nM T30085 C1LNU5 9928933 EC50 = 69 nM T30085 CKV6A4 9929398 IC50 = 1.5 nM T30085 CL1I4S 9953041 IC50 = 342 nM T30085 C38QWM 9956975 IC50 = 74000 nM T30085 CD81IB 10009210 IC50 = 371 nM T30085 C19MER 10070513 IC50 = 14 nM T30085 CC8KZ7 10073130 IC50 = 5620 nM T30085 CW10SI 10093626 IC50 = 3.7 nM T30085 C49CVF 10125816 EC50 = 190 nM T30085 CQB43I 10236901 EC50 = 510 nM T30085 CL8U9W 10301121 IC50 = 14000 nM T30085 CV32ME 10341852 IC50 = 13 nM T30085 C8WUG3 10388250 IC50 = 3090 nM T30085 CLC5R2 10431214 IC50 = 9.8 nM T30085 C9G0BJ 10431578 IC50 = 6890 nM T30085 CIV50R 10434911 IC50 = 936 nM T30085 CS1Z7H 10452736 IC50 = 30 nM T30085 CEO3K9 10453180 IC50 = 1590 nM T30085 C4XW1Y 10778685 IC50 = 51700 nM T30085 CDG74B 10806690 IC50 = 23500 nM T30085 C30MWO 10812923 IC50 = 1700 nM T30085 C9H8PW 11155568 IC50 = 50 nM T30085 C9YWX2 11166046 IC50 = 296 nM T30085 CPJ58S 11166239 IC50 = 119 nM T30085 C8ZN5I 11177436 IC50 = 28 nM T30085 CHV85J 11177940 IC50 = 52 nM T30085 C7AUJ2 11201899 IC50 = 458 nM T30085 C7NGJ8 11224807 IC50 = 491 nM T30085 CEWY62 11234901 IC50 = 132 nM T30085 C1MKF7 11236943 IC50 = 182 nM T30085 CIVK86 11259952 IC50 = 532 nM T30085 CP93BY 11282187 IC50 = 394 nM T30085 CH9IZ4 11304922 IC50 = 1.7 nM T30085 C56VGN 11305464 IC50 = 201 nM T30085 CN92CU 11328684 IC50 = 89 nM T30085 CM7Y0W 11339528 IC50 = 293 nM T30085 CTA3F7 11383983 IC50 = 66 nM T30085 CG7A2S 11385553 IC50 = 121 nM T30085 CBHX90 11396365 IC50 = 143 nM T30085 CLG02Z 11397072 IC50 = 143 nM T30085 CXDQ82 11418640 IC50 = 99 nM T30085 COPU18 11419680 EC50 = 67 nM T30085 CQ98CT 11441784 IC50 = 163 nM T30085 CXD46E 11442119 IC50 = 202 nM T30085 CG6W5A 11452732 IC50 = 121 nM T30085 C7A4HR 11454199 IC50 = 754 nM T30085 C9GFV6 11502260 IC50 = 100 nM T30085 C0IC5X 11509608 IC50 = 14 nM T30085 CE76UG 11510297 IC50 = 10 nM T30085 C2D8PW 11524511 IC50 = 8.5 nM T30085 CN28YR 11524813 IC50 = 4.8 nM T30085 C9IJ0T 11546717 IC50 = 39 nM T30085 CG0AL2 11552441 IC50 = 52 nM T30085 CN4MY1 11553111 IC50 = 19 nM T30085 C86MYU 11559484 IC50 = 49 nM T30085 C17CRP 11560307 IC50 = 8.9 nM T30085 CZ79RA 11566856 IC50 = 11 nM T30085 C7CZ8W 11596006 IC50 = 21 nM T30085 C2Q9YI 11596174 IC50 = 12 nM T30085 C8GS9Z 11646163 IC50 = 73 nM T30085 C3CY4U 11654569 IC50 = 5.2 nM T30085 C7Y0MN 11689581 IC50 = 8.3 nM T30085 CKFJ21 11703862 IC50 = 1.9 nM T30085 CN9JA5 11704217 IC50 = 180 nM T30085 CDTY94 11704386 IC50 = 9.9 nM T30085 CYK57O 11718001 IC50 = 170 nM T30085 C08ZYC 11744475 IC50 = 4700 nM T30085 C5V7SB 11749117 IC50 = 3.9 nM T30085 C3Z1HL 11750754 IC50 = 94 nM T30085 C2Y5LI 11751069 EC50 = 24 nM T30085 CTF76L 11758523 IC50 = 1730 nM T30085 C89EKZ 11949687 IC50 = 3.1 nM T30085 CIFG87 11989083 IC50 = 17.4 nM T30085 C0VF4G 12044949 IC50 = 26000 nM T30085 C5FC3A 13990811 IC50 = 18200 nM T30085 CMX78G 15979165 IC50 = 1400 nM T30085 CYT6R3 21722188 IC50 = 11.9 nM T30085 C09GWO 23581834 IC50 = 1.3 nM T30085 C7FZW6 23581843 IC50 = 7 nM T30085 C6Q4DA 23642286 IC50 = 2 nM T30085 C2L8YJ 23725183 EC50 = 2.3 nM T30085 CF1B5J 24759836 IC50 = 1.4 nM T30085 CO9J1P 24759837 EC50 = 2.8 nM T30085 C3AE6U 24764501 IC50 = 25 nM T30085 CSTE65 24768285 EC50 = 500 nM T30085 CB78ZL 24822185 IC50 = 2 nM T30085 CXBA86 24831388 IC50 = 1100 nM T30085 CD4E3U 24831389 IC50 = 620 nM T30085 CSC2K8 24831390 IC50 = 4600 nM T30085 CYH58Q 24831393 IC50 = 3600 nM T30085 C69UPX 24831712 IC50 = 45 nM T30085 CE48BP 24851760 IC50 = 5 nM T30085 C15MTU 24851762 IC50 = 5 nM T30085 C4MH7I 24851868 IC50 = 7 nM T30085 C4NLZ8 24948046 IC50 = 1.2 nM T30085 C1VP4M 24989735 IC50 = 2 nM T30085 CPC1X7 24997615 IC50 = 2.2 nM T30085 CY70QO 25099720 IC50 = 280 nM T30085 CP54GX 25099762 IC50 = 58 nM T30085 COH9F6 25168565 IC50 = 52 nM T30085 C9PYQ3 25168566 IC50 = 6 nM T30085 CA3F4Z 25168568 IC50 = 16 nM T30085 C2SLA9 25168702 IC50 = 0.3 nM T30085 CN7TU2 25168703 IC50 = 3 nM T30085 C0STB7 25168704 IC50 = 3.6 nM T30085 CDU03K 25168705 IC50 < 10 nM T30085 CZ3N7V 25168707 IC50 = 12 nM T30085 CTX09K 25168849 IC50 = 110 nM T30085 CM20EO 25168980 IC50 = 6.7 nM T30085 CT6J9S 25169379 IC50 = 1.6 nM T30085 C96QDH 25169515 IC50 = 130 nM T30085 CVWR84 25174140 IC50 = 3600 nM T30085 CE2R4Z 25197075 IC50 = 38000 nM T30085 C9E3KT 25197183 IC50 > 10000 nM T30085 CZG8J5 25197184 IC50 > 10000 nM T30085 CX1U9A 25197185 IC50 > 10000 nM T30085 CJBE59 25197291 IC50 = 5700 nM T30085 CEV78S 25197294 IC50 > 10000 nM T30085 CCW2Z3 25197296 IC50 = 6900 nM T30085 CE6U7V 25211457 IC50 = 55 nM T30085 C76CAY 25224975 IC50 = 2 nM T30085 C4FP6Y 44184119 IC50 = 7.9 nM T30085 C7E3IS 44236835 IC50 = 600 nM T30085 CS4EX5 44236837 IC50 > 1000 nM T30085 CE7A4F 44236838 IC50 > 10000 nM T30085 CI40RV 44236839 IC50 = 2500 nM T30085 C59ETX 44394297 Ki = 150 nM T30085 CJA5P8 44394328 Ki = 30 nM T30085 CWF4S2 44394360 Ki = 10 nM T30085 CKQ8C4 44394366 Ki = 20 nM T30085 COEQ58 44394379 Ki = 10 nM T30085 C1LR5Q 44394382 Ki = 30 nM T30085 CM34LN 44394389 Ki = 230 nM T30085 CAX9I5 44394395 Ki = 70 nM T30085 C4FAS7 44394396 Ki = 70 nM T30085 CHD62C 44394401 Ki = 110 nM T30085 CE95IS 44394404 Ki = 10 nM T30085 CRT40X 44394412 Ki = 80 nM T30085 CH4YD2 44394431 Ki = 9 nM T30085 C0GB3P 44394436 Ki = 20 nM T30085 CA9IK4 44394445 Ki = 40 nM T30085 CYJ6Q1 44394447 Ki > 1700 nM T30085 C0S2TF 44394455 Ki = 10 nM T30085 C20IMQ 44394486 Ki > 1700 nM T30085 CV9M5H 44394509 Ki = 1280 nM T30085 CN7A4F 44394518 Ki > 1700 nM T30085 CSRJ24 44394527 Ki = 290 nM T30085 CG6MK7 44394566 Ki = 520 nM T30085 C28OST 44405221 IC50 = 380 nM T30085 CA59JQ 44409174 IC50 = 1870 nM T30085 CPVT36 44479688 IC50 = 55 nM T30085 CWU0V2 44479689 IC50 = 180 nM T30085 C8AS2G 44479924 IC50 = 32 nM T30085 CH7I9K 44479925 IC50 = 170 nM T30085 C62WPB 44479926 IC50 = 740 nM T30085 CEO32X 44479927 IC50 = 600 nM T30085 C6H4YT 44480177 IC50 = 2400 nM T30085 C47CEW 44480436 IC50 = 36 nM T30085 C1ZC0T 44480437 IC50 = 150 nM T30085 CT4WQ2 44480438 IC50 > 30000 nM T30085 COEA34 44480439 IC50 = 590 nM T30085 CBZ3R5 44480440 IC50 > 30000 nM T30085 C3H4EV 44561635 EC50 = 970 nM T30085 CGFX45 44580555 IC50 = 33 nM T30085 CCV6U0 44580556 IC50 = 495 nM T30085 C9ODI5 44580557 IC50 = 45 nM T30085 C5RVL9 44580558 IC50 = 11000 nM T30085 CJ07PY 44580559 IC50 = 350 nM T30085 CG3WO0 44580560 IC50 = 8000 nM T30085 CN3P8S 44580561 IC50 = 15050 nM T30085 C12JQI 44580600 IC50 = 835 nM T30085 C4V8UW 44580601 IC50 = 370 nM T30085 C72UVL 44580603 IC50 = 420 nM T30085 C35GVS 44580604 IC50 = 315 nM T30085 C3NA9B 44580605 IC50 = 203 nM T30085 CU6ET7 44580606 IC50 = 430 nM T30085 C0XT7F 44580607 IC50 = 267 nM T30085 C1QM0A 44580608 IC50 = 155 nM T30085 C4J2GH 44580609 IC50 = 850 nM T30085 C8QJ0H 44580610 IC50 = 1570 nM T30085 C5EM2C 44580611 IC50 = 2000 nM T30085 C9Y0OK 44580612 IC50 = 148 nM T30085 CT51FS 44580613 IC50 = 205 nM T30085 CITM16 44580614 IC50 = 145 nM T30085 C6FY0J 44580616 IC50 = 122 nM T30085 C65HXO 44580618 IC50 = 131 nM T30085 C4L9AY 44580620 IC50 = 102 nM T30085 C3NH6G 44580622 IC50 = 154 nM T30085 CB4Z3T 44580624 IC50 = 123 nM T30085 CQTI16 44580625 IC50 = 95 nM T30085 CVYJ93 44626350 IC50 = 6.6 nM T30085 C3VT8W 44626351 IC50 = 71 nM T30085 CH2SF6 45101268 IC50 = 2.9 nM T30085 CVEI19 45101270 IC50 = 3.2 nM T30085 C98KYC 45101303 IC50 = 6.5 nM T30085 CDJ8G6 45101306 IC50 = 7.5 nM T30085 CU31BJ 45101308 IC50 = 0.8 nM T30085 C9QN4L 45101346 IC50 = 6.8 nM T30085 CN7SY1 45101347 IC50 = 2.5 nM T30085 CKY7J1 45101349 IC50 = 2.5 nM T30085 CL0GV7 45485093 IC50 = 100 nM T30085 CZ29GC 45485102 IC50 = 33 nM T30085 CZBG13 45485124 IC50 = 36 nM T30085 CB8I5E 45488012 IC50 > 1000 nM T30085 CX5B3E 45488013 IC50 = 3.8 nM T30085 CK3W2T 45488018 IC50 = 5.8 nM T30085 CX6HS7 45488023 IC50 = 2.5 nM T30085 CG1X9S 45488025 IC50 = 7.1 nM T30085 CLOC07 45488026 IC50 = 68 nM T30085 CD1R8X 45488027 IC50 > 1000 nM T30085 C4QBL8 45488028 IC50 = 70 nM T30085 CKNR92 45488030 IC50 > 1000 nM T30085 CE35BT 45488037 IC50 = 43 nM T30085 CR1OQ2 45488039 IC50 = 10 nM T30085 C7E6TD 45488040 IC50 = 100 nM T30085 C0DY9S 45488049 IC50 > 1000 nM T30085 C1XO0E 45488050 IC50 = 22 nM T30085 C1QI8N 45488053 IC50 = 100 nM T30085 CGJ30Y 45488055 IC50 = 7 nM T30085 C6SY0U 45488063 IC50 = 71 nM T30085 CB6HD1 45488064 IC50 = 1000 nM T30085 CF4O8U 45488065 IC50 = 1.3 nM T30085 CFH24W 45488067 IC50 = 13 nM T30085 C1VI8W 45488068 IC50 = 0.3 nM T30085 C2L4DC 45488083 IC50 = 0.8 nM T30085 CXQ43I 45488084 IC50 = 10 nM T30085 CI2QE1 45488087 IC50 = 8.6 nM T30085 CPCY36 46195348 IC50 = 7.5 nM T30085 CPI96D 46201936 IC50 = 32 nM T30085 CPI7Y6 46204509 IC50 = 73.6 nM T30085 C8VRT9 46204510 IC50 = 283 nM T30085 CA2T3C 46204511 IC50 = 13.4 nM T30085 C2ROV8 46204818 IC50 = 9.4 nM T30085 C16TNB 46204819 IC50 = 2.29 nM T30085 CY2R7X 46204820 IC50 = 1.77 nM T30085 CYH76W 46204821 IC50 = 37.9 nM T30085 CIR8F2 46204822 IC50 = 10.8 nM T30085 C0YOD9 46204823 IC50 = 1.68 nM T30085 CXD41T 46205138 IC50 = 1.37 nM T30085 CNBV15 46205139 IC50 = 1.78 nM T30085 CT2B4U 46205140 IC50 = 4.01 nM T30085 C48RLS 46205141 IC50 = 18.8 nM T30085 CD25IE 46205142 IC50 = 1.16 nM T30085 C9BAU2 46205143 IC50 = 1.71 nM T30085 CXGD79 46205461 IC50 = 2.68 nM T30085 CV1JB3 46205462 IC50 = 1.51 nM T30085 C87XZS 46206829 IC50 = 6.6 nM T30085 C3NO5G 46206830 IC50 = 3.4 nM T30085 CU0GS3 46206831 IC50 = 14 nM T30085 CR6C8O 46206832 IC50 = 5100 nM T30085 CK28MY 46206833 IC50 = 23 nM T30085 CKV8G1 46210599 IC50 = 25000 nM T30085 C1C8DJ 46210600 IC50 = 18000 nM T30085 C63JCQ 46228960 IC50 = 562 nM T30085 CE4OX3 46228961 IC50 = 4.06 nM T30085 C5NUB8 46228962 IC50 = 190 nM T30085 C26QUA 46228963 IC50 = 7.03 nM T30085 CF8LM1 46228977 IC50 = 17.7 nM T30085 CNC56D 46228978 IC50 = 106 nM T30085 CVM9I3 46228979 IC50 = 58.3 nM T30085 CPQM17 46228980 IC50 = 10.6 nM T30085 C25BTA 46229000 IC50 = 249 nM T30085 CNXS78 46229001 IC50 = 257 nM T30085 CT39PZ 46229002 IC50 = 119 nM T30085 C1ZXS9 46229003 IC50 = 3280 nM T30085 C15CXU 46229026 IC50 = 14.4 nM T30085 CV4L3G 46229027 IC50 = 3.51 nM T30085 CAYN51 46229028 IC50 = 762 nM T30085 CBD19Z 46229029 IC50 = 712 nM T30085 C01WRP 46229055 IC50 = 18.2 nM T30085 CD75EP 46229056 IC50 = 44.5 nM T30085 C1EOB5 46229057 IC50 = 21.8 nM T30085 CN5J0H 46229058 IC50 = 72.6 nM T30085 C9KA3V 46229086 IC50 > 10000 nM T30085 CIL3V2 46229087 IC50 > 10000 nM T30085 C4JEC9 46229153 IC50 = 1000 nM T30085 C01HGP 46229154 IC50 = 7000 nM T30085 CN1B9F 46229155 IC50 = 35000 nM T30085 C1J7NT 46229156 IC50 = 11000 nM T30085 COF9A7 46229157 IC50 = 1000 nM T30085 CEI97D 46229158 IC50 = 78000 nM T30085 C0NE3T 46229159 IC50 = 12000 nM T30085 CPO40S 46229160 IC50 > 100000 nM T30085 CS61BK 46229176 IC50 = 6910 nM T30085 CND7T4 46229177 IC50 > 10000 nM T30085 CC3PN5 46229188 IC50 = 1420 nM T30085 CNQ9V3 46229189 IC50 = 1230 nM T30085 CIW82T 46229190 IC50 = 542 nM T30085 CJQ24G 46229191 IC50 = 103 nM T30085 C8C2RN 46229215 IC50 = 24.9 nM T30085 CP53XV 46229216 IC50 = 45.3 nM T30085 CZ8OI5 46229217 IC50 = 53 nM T30085 C7R8XA 46229218 IC50 = 2390 nM T30085 C2LX1N 46229237 IC50 > 10000 nM T30085 CFSJ29 46229238 IC50 = 214 nM T30085 C4W6BN 46229239 IC50 = 379 nM T30085 C62QNC 46229240 IC50 = 353 nM T30085 CF51PZ 46229264 IC50 = 122 nM T30085 C02CZL 46229265 IC50 = 146 nM T30085 C23ERB 46229266 IC50 = 10.9 nM T30085 CG6I8X 46229267 IC50 = 155 nM T30085 CM5G2B 46229268 IC50 = 758 nM T30085 CQZ0M9 46229292 IC50 = 445 nM T30085 CEI20F 46229293 IC50 = 16.6 nM T30085 CZTS95 46229294 IC50 = 126 nM T30085 CX92KB 46229295 IC50 = 30.3 nM T30085 CM2R3J 46229314 IC50 = 638 nM T30085 CLF4M1 46229315 IC50 = 97.4 nM T30085 CL7FB3 46229316 IC50 = 36.4 nM T30085 C5V2WF 46229317 IC50 = 81.6 nM T30085 CJ61SL 46861619 IC50 = 74 nM T30085 C4IP5Z 46865788 IC50 = 3 nM T30085 CG50FN 46865896 IC50 = 7.9 nM T30085 CV7D4P 46881659 IC50 = 1000 nM T30085 CC21VE 46881660 IC50 > 10000 nM T30085 CPUY71 46881661 IC50 = 140 nM T30085 CP3OQ5 46881662 IC50 = 2000 nM T30085 CDMF67 46881707 IC50 = 3700 nM T30085 C1XW5V 46881708 IC50 = 139 nM T30085 CQ04HT 46881709 IC50 = 2.4 nM T30085 CLFM76 46881760 IC50 = 5.1 nM T30085 C4EQH7 46881761 IC50 = 59 nM T30085 CI9VO5 46881762 IC50 = 53 nM T30085 C03QUF 46889407 IC50 = 202 nM T30085 C0PN8T 46889427 IC50 = 43 nM T30085 C6ZU7V 46889428 IC50 = 70.8 nM T30085 CXT6D1 46889429 IC50 = 110 nM T30085 C4N8RH 46889430 IC50 = 109 nM T30085 C7WN2K 46889431 IC50 = 435 nM T30085 CJ71LZ 46889455 IC50 = 17 nM T30085 CBI75R 46889456 IC50 = 17.3 nM T30085 C2LKX8 46889457 IC50 = 111 nM T30085 C4QXM2 46889458 IC50 = 77.6 nM T30085 C4CZS2 46889467 IC50 = 13.4 nM T30085 C5YDZ8 46889468 IC50 = 71.3 nM T30085 CNRH61 46889469 IC50 = 1870 nM T30085 CX6V0W 46889470 IC50 = 293 nM T30085 CDYS29 46889471 IC50 = 131 nM T30085 CWAM21 46889644 IC50 = 237 nM T30085 CQ86JT 46889645 IC50 = 259 nM T30085 C8V5HF 46889646 IC50 = 356 nM T30085 C2MQK0 46889647 IC50 = 811 nM T30085 C4CDL2 46889648 IC50 = 134 nM T30085 CP3UX0 46889671 IC50 = 176 nM T30085 CDXG93 46889672 IC50 = 64.3 nM T30085 CML08C 46889673 IC50 = 61.3 nM T30085 C8D7IO 46889674 IC50 = 71.4 nM T30085 C6EH8N 46889702 IC50 = 75.4 nM T30085 CVE39O 46889703 IC50 = 168 nM T30085 CE9A0N 46889704 IC50 = 222 nM T30085 CXD7Q8 46889705 IC50 = 272 nM T30085 CR5V4F 46889731 IC50 = 351 nM T30085 CD8QG7 46889732 IC50 = 64.9 nM T30085 CDP5C2 46889733 IC50 = 82.7 nM T30085 CWPT61 46889734 IC50 = 103 nM T30085 C2NPM7 46889773 IC50 = 11.4 nM T30085 CCF3K7 46889774 IC50 = 1710 nM T30085 CN7R3T 46889775 IC50 = 700 nM T30085 C5X6WH 46889776 IC50 = 1140 nM T30085 CR46NU 46889813 IC50 = 1040 nM T30085 C7XI8J 46889814 IC50 = 1520 nM T30085 CY4BM6 46889815 IC50 = 10000 nM T30085 C4EM8B 46889816 IC50 = 10000 nM T30085 C39CJH 46897476 IC50 = 81 nM T30085 C6Q0NU 46897565 IC50 = 322 nM T30085 C1CZ4A 46897566 IC50 = 20 nM T30085 CRF28B 46897567 IC50 = 26 nM T30085 C5UWM8 46897656 IC50 = 28 nM T30085 C7OW4N 46897658 IC50 = 64 nM T30085 CMGI18 46906366 IC50 = 0.9 nM T30085 CF2K6T 46906391 IC50 = 170 nM T30085 C6JKR2 46906469 IC50 = 0.9 nM T30085 C3WJN0 46927885 IC50 = 121 nM T30085 CWR0G5 49863594 IC50 = 610 nM T30085 CO09GW 49863595 IC50 > 10000 nM T30085 CJ14CV 49863596 IC50 = 4630 nM T30085 CIVP10 49863597 IC50 > 10000 nM T30085 CN1CM5 49863623 IC50 > 10000 nM T30085 CES3L5 49863624 IC50 > 10000 nM T30085 CQY76J 49863625 IC50 > 10000 nM T30085 CBP54H 49863626 IC50 > 10000 nM T30085 CE1H4C 49863627 IC50 > 10000 nM T30085 CGUD90 49863655 IC50 = 1050 nM T30085 CL6KO3 49863656 IC50 = 786 nM T30085 CP9MK4 49863657 IC50 = 2360 nM T30085 C23QLI 49863658 IC50 = 8640 nM T30085 C4DBL0 49863659 IC50 = 257 nM T30085 CO3Z7V 49863696 IC50 = 251 nM T30085 CIA85L 49863697 IC50 = 411 nM T30085 CRV61E 50925634 EC50 = 161 nM T30085 C30UZQ 50942027 IC50 = 19.8 nM T30085 CBZW98 50992816 EC50 = 12915 nM T30085 C0VDU9 50992817 EC50 = 893 nM T30085 C6SP8V 50992818 EC50 = 275 nM T30085 C28ESY 50992819 EC50 = 1161 nM T30085 C7Y2IX 50992875 EC50 = 255 nM T30085 CGN81J 50992876 EC50 = 241 nM T30085 C7FIY3 50993229 EC50 = 7129 nM T30085 C0BZ4A 50993230 EC50 = 1094 nM T30085 CH2M5L 50993298 EC50 = 40589 nM T30085 CGVD67 50993299 EC50 = 3033 nM T30085 C60VQY 50993300 EC50 = 12956 nM T30085 CUN37X 50993301 EC50 = 2237 nM T30085 CUV37C 50993302 EC50 = 12415 nM T30085 C5EY8X 50993303 EC50 = 23627 nM T30085 CRF1J3 50993304 EC50 = 9821 nM T30085 CN85YV 50993373 EC50 = 865 nM T30085 C8WI1H 50993374 EC50 = 28217 nM T30085 C1GO3Z 50993375 EC50 = 10279 nM T30085 C0HB2X 50993376 EC50 = 10680 nM T30085 CMR3S6 50993377 EC50 = 923 nM T30085 CN9BV1 50993378 EC50 = 1819 nM T30085 CQF19B 50993379 EC50 = 5487 nM T30085 CFRQ51 50993456 EC50 > 50000 nM T30085 C28TGC 50993457 EC50 = 8600 nM T30085 C42OVM 50993628 EC50 = 1376 nM T30085 CZO27N 50993629 EC50 = 30931 nM T30085 CFG4E8 50993630 EC50 = 473 nM T30085 CL4R9S 50993631 EC50 = 1288 nM T30085 C8MA4B 50993632 EC50 = 1410 nM T30085 CY4JG3 50993633 EC50 = 11137 nM T30085 CD3N4X 50993708 EC50 = 297 nM T30085 C3XDO5 50993709 EC50 = 1682 nM T30085 CZ5AB3 50993710 EC50 = 633 nM T30085 C09SZJ 50993711 EC50 = 863 nM T30085 C2XLV3 50993712 EC50 = 233 nM T30085 C4YF1K 50993787 EC50 = 426 nM T30085 C6A9SK 50993788 EC50 = 1334 nM T30085 CKS3C8 50993789 EC50 = 530 nM T30085 CPR0Q8 50993790 EC50 = 577 nM T30085 CR4MT3 51003384 IC50 = 0.72 nM T30085 C0HC4A 51346777 IC50 = 0.772 nM T30085 C9VI3M 52918252 IC50 = 9 nM T30085 C1AE6L 52918253 IC50 = 10 nM T30085 C75QOX 52940815 IC50 = 17 nM T30085 CDPR75 52940816 IC50 = 32 nM T30085 CFOA48 52940817 IC50 = 8.1 nM T30085 CXV49H 52941153 IC50 = 73.6 nM T30085 CZ4U6T 52941464 IC50 = 119 nM T30085 C5YCL8 52942697 IC50 = 8870 nM T30085 CC3Q0A 52942925 IC50 = 246 nM T30085 C5HF7S 52943562 IC50 = 107 nM T30085 CZW76K 52943577 IC50 = 34.5 nM T30085 CWYB57 52943591 IC50 = 17.1 nM T30085 CQHI10 52943615 IC50 = 39.4 nM T30085 C27WTS 52943956 IC50 = 447 nM T30085 CLF61E 52943983 IC50 = 76 nM T30085 C3X1MP 52944051 IC50 = 2.2 nM T30085 C5GLF2 52944790 IC50 = 36.8 nM T30085 CEC92L 52945162 IC50 = 189 nM T30085 CE8S4W 52946050 IC50 = 10.7 nM T30085 C8LJT3 52946381 IC50 = 223 nM T30085 CA7U8W 52946416 IC50 = 130 nM T30085 CGW25J 52947271 IC50 = 64.4 nM T30085 C0CES2 52947478 IC50 = 124 nM T30085 CMV2G0 52948079 IC50 = 920 nM T30085 C4G7CR 52949327 IC50 = 28 nM T30085 CK9R5G 52949970 IC50 = 113 nM T30085 C1Z2BC 52950032 IC50 = 46.9 nM T30085 CPN62X 52950124 IC50 = 2.4 nM T30085 C7BDP8 53317204 IC50 = 68.9 nM T30085 C9ZW4L 53317310 IC50 = 18.6 nM T30085 C7X4JZ 53317450 IC50 = 5 nM T30085 CD6LJ4 53317451 IC50 = 18.8 nM T30085 CPB3I1 53317452 IC50 = 12.4 nM T30085 CK25BG 53317453 IC50 = 14 nM T30085 CP6ZE5 53318597 IC50 = 7.01 nM T30085 CTU85W 53318598 IC50 = 20.8 nM T30085 CVQS75 53318599 IC50 = 23.5 nM T30085 C6J0PE 53318600 IC50 = 89.5 nM T30085 C15CNQ 53318726 IC50 = 21.2 nM T30085 CPG56Z 53318727 IC50 = 6.11 nM T30085 CGA7R0 53318728 IC50 = 7.36 nM T30085 C1NTD9 53318729 IC50 = 4.47 nM T30085 CLY1J6 53319918 IC50 = 10.6 nM T30085 C9N2PJ 53319919 IC50 = 68.7 nM T30085 C6EA0K 53320039 IC50 = 25.4 nM T30085 C2IYC1 53320040 IC50 = 8.2 nM T30085 CX8W3B 53320041 IC50 = 56.4 nM T30085 CJ3CE9 53320042 IC50 = 18.9 nM T30085 C12XAP 53320043 IC50 = 1.57 nM T30085 C36MLO 53320044 IC50 = 1.28 nM T30085 C6TJ5Q 53320045 IC50 = 1.89 nM T30085 C1SW5E 53320046 IC50 = 6.36 nM T30085 C3U2NG 53320047 IC50 = 9.73 nM T30085 CP49LD 53320048 IC50 = 1.11 nM T30085 CLO64C 53321224 IC50 = 54.9 nM T30085 CZLA75 53321225 IC50 = 1450 nM T30085 CO0HM1 53321352 IC50 = 13.3 nM T30085 CY8HQ1 53321353 IC50 = 58.7 nM T30085 CA3WI0 53321354 IC50 > 10000 nM T30085 CC73LO 53321355 IC50 = 1.43 nM T30085 C52PND 53321356 IC50 = 140 nM T30085 C2R4DE 53321425 IC50 = 54.8 nM T30085 C7RTN9 53321426 IC50 = 31.9 nM T30085 C7LYR8 53321459 IC50 = 16.7 nM T30085 CR95VK 53321598 IC50 = 471 nM T30085 CF7Q1C 53321704 IC50 = 48.9 nM T30085 C6VB9G 53322674 IC50 = 119 nM T30085 C1UAN4 53322675 IC50 = 13.3 nM T30085 CH58CT 53322676 IC50 = 22.6 nM T30085 CI1D0X 53322677 IC50 = 1.42 nM T30085 CCF5O8 53323798 IC50 = 106 nM T30085 CVU0W5 53323877 IC50 = 59.1 nM T30085 C61QHF 53324010 IC50 = 9.71 nM T30085 C5M8EX 53324011 IC50 = 19.6 nM T30085 C0EW8G 53324012 IC50 = 13.3 nM T30085 CL48AO 53324013 IC50 = 2.79 nM T30085 C4QZY9 53325167 IC50 = 110 nM T30085 CV41LH 53325311 IC50 = 51.4 nM T30085 C7NJO1 53325312 IC50 = 4.69 nM T30085 CP38HM 53325313 IC50 = 11.5 nM T30085 C2GVS4 53325314 IC50 = 1.14 nM T30085 C5XVR7 53325315 IC50 = 3.13 nM T30085 C23AWE 53325316 IC50 = 14.6 nM T30085 COH1T6 53325317 IC50 = 36.7 nM T30085 C8W6EB 53326413 IC50 = 156 nM T30085 C27PUZ 53326458 IC50 = 13.5 nM T30085 CTC3B7 53326459 IC50 = 23.8 nM T30085 CMS5X4 53326460 IC50 = 9.55 nM T30085 CV2A4I 53326576 IC50 = 12.4 nM T30085 C0N6OP 53326577 IC50 = 30.9 nM T30085 CH5US7 53326578 IC50 = 9.31 nM T30085 C71UIW 53326797 IC50 = 30.9 nM T30085 CXA5I2 53326894 IC50 = 50.3 nM T30085 CF93AV 53326940 IC50 = 54.8 nM T30085 CXQ43D 53327912 IC50 = 0.934 nM T30085 CJ9C1N 53327913 IC50 = 0.797 nM T30085 CL90ZJ 53328104 IC50 = 1.59 nM T30085 CF3Q2T 53328105 IC50 = 1.29 nM T30085 CKB6T4 53328106 IC50 = 2.01 nM T30085 CA86TE 53328107 IC50 = 6.08 nM T30085 CL4C0K 53328108 IC50 = 3.98 nM T30085 CP3Z7X 53328109 IC50 = 4.35 nM T30085 CQM91N 53328306 IC50 = 4.29 nM T30085 CI2L5S 53328307 IC50 = 1.18 nM T30085 C2YQ1S 53328308 IC50 = 2.87 nM T30085 CY9C6D 53328309 IC50 = 7.55 nM T30085 CFI51G 53328310 IC50 = 1.24 nM T30085 C8DLU2 53328498 IC50 = 1.54 nM T30085 CX8U6I 53328499 IC50 = 1.69 nM T30085 C78ATU 53328500 IC50 = 3.38 nM T30085 CS5A1R 53328501 IC50 = 4.22 nM T30085 CLUW49 53328502 IC50 = 21.6 nM T30085 C1N9MZ 53328679 IC50 = 2.23 nM T30085 CGHS20 53328680 IC50 = 32.8 nM T30085 CR97SY 53328681 IC50 = 1.51 nM T30085 CK6D4C 53328682 IC50 = 5.55 nM T30085 CFD7R6 53328683 IC50 = 131 nM T30085 C2T4EM 53328863 IC50 = 713 nM T30085 CN49HA 53328864 IC50 = 5.81 nM T30085 C6HT8K 53328865 IC50 = 20.5 nM T30085 CHC04P 53328866 IC50 = 5.88 nM T30085 CUNA45 53328867 IC50 = 2.23 nM T30085 CCM6S3 53329034 IC50 = 17.5 nM T30085 CU1Q7X 53329035 IC50 = 38.7 nM T30085 CLE0P6 53329036 IC50 = 16.2 nM T30085 CMUT30 53329037 IC50 = 10 nM T30085 CM7BV1 53329038 IC50 = 3.49 nM T30085 CO79TC 53329218 IC50 = 5.35 nM T30085 CL0MW1 53329219 IC50 = 3.88 nM T30085 CKZ13A 53329220 IC50 = 2.12 nM T30085 CU1X8P 53329221 IC50 = 4.57 nM T30085 CJ9KA5 53329222 IC50 = 27.4 nM T30085 C9IKL8 53329223 IC50 = 2.24 nM T30085 CM6T5Q 53329400 IC50 = 13.3 nM T30085 CZ4D6B 53329401 IC50 = 4.77 nM T30085 CRAW58 53329402 IC50 = 2.31 nM T30085 CDQ2T1 53330783 IC50 = 2.15 nM T30085 C8IS9P 53330784 IC50 = 7.37 nM T30085 CR1B2U 53363121 IC50 > 1000 nM T30085 CMW1K2 53363122 IC50 = 680 nM T30085 CFJ5G8 53389526 IC50 = 12 nM T30085 CVR7K0 53467552 IC50 = 83 nM T30085 CVL86S 53467553 IC50 = 120 nM T30085 C2ED6O 53467554 IC50 = 252 nM T30085 CW40YV 53467555 IC50 = 89 nM T30085 CX7P2D 53467556 IC50 = 762 nM T30085 C5YX0V 53467759 IC50 = 141 nM T30085 C8CLN9 53467761 IC50 = 80 nM T30085 C7Q6AJ 53467762 IC50 = 110 nM T30085 C92DHW 53467763 IC50 = 107 nM T30085 C6O3NH 53467764 IC50 = 222 nM T30085 C0T5VA 53467975 IC50 = 33 nM T30085 C78TRY 53468202 IC50 = 23.6 nM T30085 C2N8AH 53468203 IC50 = 248 nM T30085 C7VQG5 53468204 IC50 = 489 nM T30085 C2XHO3 53468206 IC50 = 10.9 nM T30085 C31UEL 53468414 IC50 = 328 nM T30085 C27COD 53472857 IC50 = 1.38 nM T30085 CWKO38 53494878 IC50 = 0.899 nM T30085 COG65P 53494879 IC50 = 2.27 nM T30085 C1NJ5P 54579981 IC50 = 150 nM T30085 CL4K3S 54579982 IC50 = 30 nM T30085 CLMR05 54580869 IC50 = 59 nM T30085 C0S2FU 54580870 IC50 = 73 nM T30085 CQB85M 54580871 IC50 = 13 nM T30085 CW1HF3 54580872 IC50 = 3 nM T30085 CMV2C5 54580873 IC50 = 12 nM T30085 C85GSF 54580894 IC50 = 10 nM T30085 CAL4P2 54580976 IC50 = 40 nM T30085 CZ0MV1 54580977 IC50 = 70 nM T30085 CN84QS 54581929 IC50 = 89 nM T30085 CMXZ95 54581951 IC50 = 4 nM T30085 CLJ76E 54581991 IC50 = 1100 nM T30085 CYW6B8 54581992 IC50 = 250 nM T30085 C0QA6R 54582021 IC50 = 1580 nM T30085 C0IC6L 54582851 IC50 = 36 nM T30085 CD7M2S 54582852 IC50 = 21 nM T30085 CC7AP2 54582873 IC50 = 5100 nM T30085 C1N0KC 54582874 IC50 = 5 nM T30085 CP8L4K 54582928 IC50 = 370 nM T30085 COS5F2 54582929 IC50 = 2100 nM T30085 CO82HW 54582930 IC50 = 150 nM T30085 CJ6WB3 54582969 IC50 = 640 nM T30085 C46EPV 54582970 IC50 = 180 nM T30085 CM8PX5 54583110 EC50 = 1.1 nM T30085 C9TY5S 54583857 IC50 = 9800 nM T30085 C9A2QD 54583858 IC50 = 23 nM T30085 C5EPU2 54583960 IC50 = 160 nM T30085 CB6Z4P 54584816 IC50 = 480 nM T30085 CNB69R 54584817 IC50 = 8 nM T30085 CSH0W9 54584818 IC50 = 10 nM T30085 CZ1P6F 54584819 IC50 = 41 nM T30085 CV2R1U 54584874 IC50 = 2110 nM T30085 CLH1P6 54584875 IC50 = 80 nM T30085 C7KRD4 54584876 IC50 = 520 nM T30085 C39LNR 54585760 IC50 = 10000 nM T30085 C7LQ4K 54585761 IC50 = 22 nM T30085 CP53UO 54585762 IC50 = 660 nM T30085 CC2F5M 54585763 IC50 = 13 nM T30085 CHFT12 54585791 IC50 = 3 nM T30085 C5W0CS 54585841 IC50 = 1200 nM T30085 CNIF43 54585871 IC50 = 30 nM T30085 COGZ89 54586754 IC50 = 57 nM T30085 CEU21Q 54586755 IC50 = 7 nM T30085 C1MTS5 54586771 IC50 = 110 nM T30085 CLM0E5 54586807 IC50 = 90 nM T30085 C0A1GD 54586808 IC50 = 430 nM T30085 CV8LG7 54587778 IC50 = 14 nM T30085 CJ3P7X 54587797 IC50 = 7 nM T30085 CILJ80 54587798 IC50 = 5 nM T30085 CWAK94 54587799 IC50 = 8 nM T30085 C4RI6X 54597681 IC50 = 4.47 nM T30085 CUWV29 54597682 IC50 = 12.4 nM T30085 CSD4P1 54597683 IC50 = 8.73 nM T30085 CT4RA9 56658254 IC50 = 1.35 nM T30085 CSP37N 56658255 IC50 = 0.778 nM T30085 C7B9KY 56659829 IC50 > 10000 nM T30085 CZ79IH 56659854 IC50 = 69.6 nM T30085 C4E5DX 56659941 IC50 = 10.3 nM T30085 C5I8QS 56659942 IC50 = 91.3 nM T30085 CSE1K8 56661751 IC50 = 3.65 nM T30085 CTVO72 56661752 IC50 = 1.38 nM T30085 CG9B5C 56663408 IC50 = 162 nM T30085 C5KW2N 56663480 IC50 = 34.6 nM T30085 CJ6E7M 56663481 IC50 = 54.6 nM T30085 C3JPH9 56666658 IC50 > 10000 nM T30085 CJ6HG9 56666748 IC50 = 49.5 nM T30085 C0W9YH 56666838 IC50 = 94 nM T30085 CL24PM 56666839 IC50 = 11.9 nM T30085 CBM98W 56668635 IC50 = 1.34 nM T30085 CPE73B 56668636 IC50 = 1.59 nM T30085 C3NSO7 56670145 IC50 > 10000 nM T30085 CLQ75X 56670174 IC50 = 88.3 nM T30085 CKTX60 56670175 IC50 = 29.3 nM T30085 CD7Q4N 56670266 IC50 = 115 nM T30085 C97OWV 56670267 IC50 = 60.2 nM T30085 C0Q5JG 56670358 IC50 = 140 nM T30085 C6EXT3 56672119 IC50 = 2.95 nM T30085 CT9FS1 56672120 IC50 = 0.974 nM T30085 CI68XQ 56672121 IC50 = 1.4 nM T30085 CMA48J 56673660 IC50 > 10000 nM T30085 C6HKW4 56673661 IC50 > 1000 nM T30085 CC5X9D 56673698 IC50 = 21.1 nM T30085 CAME43 56673699 IC50 = 71.4 nM T30085 CS3QZ4 56673700 IC50 = 68.9 nM T30085 CNA7V1 56673701 IC50 = 59.8 nM T30085 CMA06D 56675515 IC50 = 3.63 nM T30085 CUJ7D1 56675519 IC50 = 1.4 nM T30085 CTL9A8 56676982 IC50 = 9000 nM T30085 CT75KO 56677009 IC50 = 50.2 nM T30085 C3AH7S 56677111 IC50 = 48.4 nM T30085 CVB0O1 56677129 IC50 = 86.5 nM T30085 CJT7E1 56677187 IC50 = 65 nM T30085 CMX43I 56680163 IC50 > 100000 nM T30085 C1O9BE 56680435 IC50 = 12.8 nM T30085 C32HVL 56680436 IC50 = 57.2 nM T30085 C3M4KL 56680495 IC50 = 11.5 nM T30085 C1MT3N 56683501 IC50 > 10000 nM T30085 CKN06T 56683502 IC50 > 1000 nM T30085 CR0L1D 56683663 IC50 = 27.5 nM T30085 CC7G0L 56683664 IC50 = 451 nM T30085 CSY83X 56683665 IC50 = 24.8 nM T30085 C2X5JK 56683756 IC50 = 70.7 nM T30085 C40RPD 56683828 IC50 = 111 nM T30085 C3PXR7 56928196 Ki = 1.1 nM T30085 C34PBD 56942482 IC50 = 17 nM T30085 C7M0QO 57556376 IC50 = 16.8 nM T30085 CPS65X 57556380 IC50 = 122.7 nM T30085 C7E8MR 57556391 IC50 = 3.2 nM T30085 CJ59CN 57556398 IC50 = 3.6 nM T30085 CP82CI 57556406 IC50 = 7.5 nM T30085 CIL8S9 57556409 IC50 = 14.2 nM T30085 CUL1T8 57556416 IC50 = 1.4 nM T30085 C9OW3L 57556425 IC50 = 9.1 nM T30085 CZ5B2H 57556428 IC50 = 14.5 nM T30085 CL52JF 57556430 IC50 = 29.9 nM T30085 CF70BA 57556431 IC50 = 117.9 nM T30085 CO01YH 57556433 IC50 = 4.8 nM T30085 C5IY8V 57802355 IC50 = 377 nM T30085 CZ9N7D 57802433 IC50 = 231 nM T30085 CTA1V4 58178431 IC50 = 18000 nM T30085 C2VP8M 58186566 IC50 = 7.1 nM T30085 CQ1RO6 58239014 IC50 = 3 nM T30085 C4IS2L 58242596 IC50 = 381 nM T30085 C6I4LS 58507570 IC50 = 1.4 nM T30085 CJ14PC 58786124 IC50 = 44000 nM T30085 C0T2FG 58786126 IC50 = 12000 nM T30085 CWK40A 58786134 IC50 = 5200 nM T30085 C85JXA 58786137 IC50 = 970 nM T30085 C40NPF 58786147 IC50 = 39 nM T30085 CR6SN3 58786158 IC50 = 99 nM T30085 CH39MN 58786180 IC50 = 16 nM T30085 CEP39H 58786231 IC50 = 17 nM T30085 C04JZV 58843397 IC50 = 92 nM T30085 CK2F7O 58843413 IC50 = 2300 nM T30085 C8MW1U 58843421 IC50 = 675 nM T30085 CY7TA8 58843422 IC50 > 100000 nM T30085 CN2O8L 58843447 IC50 = 4900 nM T30085 C3C2NK 58843468 IC50 = 650 nM T30085 CG1VX7 58843469 IC50 = 75 nM T30085 C7Z8IB 58843499 IC50 = 610 nM T30085 C7VZQ4 58843539 IC50 > 100000 nM T30085 CYUM37 58843551 IC50 > 100000 nM T30085 C8DJ2C 58843565 IC50 = 6300 nM T30085 C31JST 58843616 IC50 = 47 nM T30085 C0C9PL 59740011 IC50 = 1.1 nM T30085 CH4JP5 60134927 IC50 = 1.6 nM T30085 C3QB7A 66608038 IC50 = 7.3 nM T30085 C4AHP2 66691967 IC50 = 15800 nM T30085 CPB6R3 67196949 IC50 = 1.6 nM T30085 C0IAX7 67198213 IC50 = 69 nM T30085 C9R4CE 67199199 IC50 = 1098 nM T30085 CHS7E9 67304774 IC50 = 4 nM T30085 C5XP9B 67891757 IC50 = 0.67 nM T30085 CAM0S1 68535905 IC50 = 46 nM T30085 C6XLO5 68537281 IC50 = 151 nM T30085 CIOM04 68538795 IC50 = 20 nM T30085 CU2YH4 68538810 IC50 = 608 nM T30085 CY9W4S 68538834 IC50 = 1050 nM T30085 CCP3K5 68540044 IC50 = 209 nM T30085 CHS98N 68540709 IC50 = 1070 nM T30085 C02MEL 68542200 IC50 = 80 nM T30085 CS3BC9 69516549 IC50 = 75900 nM T30085 C0AS6H 69516684 IC50 = 13900 nM T30085 CMB3H2 69516839 IC50 = 64700 nM T30085 CF50GR 69624867 IC50 = 0.8 nM T30085 C02YNI 70684428 EC50 = 3632 nM T30085 C3TL7D 70684429 EC50 = 47 nM T30085 CNM2G0 70686571 EC50 = 151 nM T30085 CDH53P 70688690 EC50 = 25505 nM T30085 C5SRW9 70690752 EC50 = 588 nM T30085 C4CK1J 70691761 IC50 = 100 nM T30085 CDR2S1 70692889 EC50 = 1110 nM T30085 COFW37 70692890 EC50 = 87 nM T30085 CLSI96 70692891 EC50 = 50 nM T30085 C47OBZ 70694930 EC50 = 4153 nM T30085 C35JTP 70695943 IC50 = 70 nM T30085 CX13VG 70696980 EC50 = 736 nM T30085 C84IFU 70696981 EC50 = 722 nM T30085 CC9AH0 71451518 IC50 = 60500 nM T30085 CV7Y2F 71453231 IC50 = 7 nM T30085 CG9TO4 71453232 IC50 = 6010 nM T30085 CB6Z5A 71453233 IC50 = 5980 nM T30085 C07IRW 71453345 IC50 = 14100 nM T30085 C54QMZ 71454958 IC50 = 156000 nM T30085 C3LBY4 71454959 IC50 = 5010 nM T30085 C2BOR8 71454960 IC50 = 5680 nM T30085 CL5P0D 71454961 IC50 = 154 nM T30085 CZ6QB5 71454962 IC50 = 68 nM T30085 C61YGV 71455054 IC50 = 1390 nM T30085 CA1SU7 71455055 IC50 = 2020 nM T30085 CHGR43 71456753 IC50 = 2790 nM T30085 CDJ14N 71456754 IC50 = 3580 nM T30085 C6DRB5 71456755 IC50 = 285 nM T30085 CE6F9D 71457086 IC50 = 240.8 nM T30085 C3DN7L 71458597 IC50 = 14900 nM T30085 CZWO59 71460439 IC50 = 4140 nM T30085 C69OZJ 71460532 IC50 = 204000 nM T30085 C7DMG8 71462125 IC50 = 13300 nM T30085 CMG4Y3 71462176 IC50 = 65700 nM T30085 CA6VK1 71462236 IC50 = 18500 nM T30085 CT73OL 71524007 IC50 = 5100 nM T30085 CM2LH3 71524008 IC50 = 3980 nM T30085 CH9SD8 71524009 IC50 = 2470 nM T30085 CX4Q0G 71524030 IC50 = 9950 nM T30085 C3E9IM 71524031 IC50 = 2540 nM T30085 C4IBY1 71524032 IC50 = 457 nM T30085 COGI16 71524033 IC50 = 358 nM T30085 CH96ZJ 71524034 IC50 = 319 nM T30085 CEZ71U 71524035 IC50 = 8 nM T30085 CRC40T 71524036 IC50 = 18 nM T30085 CX8U3Q 71524037 IC50 = 42 nM T30085 CA1I2V 71524038 IC50 = 98 nM T30085 C70ITO 71603300 EC50 = 39 nM T30085 CR4IJ0 71603301 EC50 = 3441 nM T30085 CR8M7J 71604141 EC50 = 92 nM T30085 CHS89O 71604142 EC50 = 88 nM T30085 CBG14D 71604199 EC50 = 63 nM T30085 C8S1NV 71604200 EC50 = 175 nM T30085 CQ3T0D 71604202 EC50 = 130 nM T30085 CL7R1O 71604268 EC50 = 65 nM T30085 C4G6DV 71604269 EC50 = 38 nM T30085 CZTA53 71604270 EC50 = 42 nM T30085 C4MB1Y 71713605 IC50 = 70 nM T30085 CCF8L3 71713606 IC50 = 14 nM T30085 CDN34F 71770704 IC50 = 1 nM T30085 COA62F 71770819 IC50 = 2.4 nM T30085 CE6QS8 71770820 IC50 = 1.5 nM T30085 C2YSN9 72192599 IC50 = 163 nM T30085 C9Z6FI 72192600 IC50 = 6671 nM T30085 CX0UM3 73346536 EC50 = 2500 nM T30085 CJ01LN 73348014 EC50 = 34000 nM T30085 C7GCY0 73348015 EC50 = 620 nM T30085 C47OTD 73348016 EC50 > 50000 nM T30085 CZ9AT7 73348017 EC50 = 3700 nM T30085 CTDC49 73348018 EC50 > 50000 nM T30085 CFC4W1 73349554 EC50 > 50000 nM T30085 C2R0ZL 73349555 EC50 = 24000 nM T30085 CS97BC 73354077 EC50 = 11000 nM T30085 CKC2V7 73354078 EC50 = 21000 nM T30085 CYWE90 73354079 EC50 = 35000 nM T30085 CD9T0X 73354080 EC50 > 50000 nM T30085 CU0Z8P 73354081 EC50 = 5100 nM T30085 C9SZN5 73355608 EC50 = 33000 nM T30085 CW8XK6 73357149 EC50 = 46000 nM T30085 C56WLN 73357150 EC50 > 50000 nM T30085 C8QFY5 73357151 EC50 > 50000 nM T30085 CNX4Y8 74538678 IC50 = 2.5 nM T30085 CUI04H 76070792 IC50 = 1.9 nM T30085 C65ICL 76070894 IC50 = 2.7 nM T30085 CC4U0L 76070897 IC50 = 3.6 nM T30085 C5TP1J 76070999 IC50 = 4.3 nM T30085 CCL50G 76071000 IC50 = 0.9 nM T30085 C60BEU 76071231 IC50 = 5.2 nM T30085 C65CMH 76310235 IC50 = 18 nM T30085 CMIF39 76310883 IC50 = 134.7 nM T30085 C5LZ9K 76310884 IC50 = 163.2 nM T30085 CA85TN 76313928 IC50 = 2.2 nM T30085 C21SOA 76314516 IC50 = 146.9 nM T30085 CE4MR2 76315186 IC50 = 34100 nM T30085 CYVA36 76317461 IC50 = 11 nM T30085 CPF3Q2 76318092 IC50 = 367 nM T30085 CX2H5F 76318093 IC50 = 311 nM T30085 CL2WO9 76321790 IC50 = 214.2 nM T30085 CE07JZ 76325427 IC50 = 185.8 nM T30085 CEKB95 76325428 IC50 = 175 nM T30085 C1ZP0V 76325429 IC50 = 458 nM T30085 C82SWJ 76325430 IC50 = 149.1 nM T30085 CM79IF 76328370 IC50 = 93 nM T30085 CF0R6P 76328964 IC50 = 190.3 nM T30085 C2T7KO 76332640 IC50 = 227 nM T30085 CO67AZ 76335657 IC50 = 24 nM T30085 CXH87A 76336244 IC50 = 150 nM T30085 CLV1N4 76336245 IC50 = 151.8 nM T30085 C2G4YS 76336246 IC50 = 125.9 nM T30085 C4RY1I 86282875 IC50 = 1.3 nM T30085 C2ZMG1 89630294 EC50 = 237 nM T30085 CTN7F4 89630298 EC50 = 359 nM T30085 COM9Z6 89630299 EC50 = 1585 nM T30085 CES8X4 89630301 EC50 = 552 nM T30085 CI17QE 89630302 EC50 = 113 nM T30085 CC45KG 89630303 EC50 = 499 nM T30085 CVU08Y 89630305 EC50 = 160 nM T30085 CLI2R9 89630307 EC50 = 387 nM T30085 C7U8EF 89630310 EC50 = 151 nM T30085 C1EU9Y 89630311 EC50 = 716 nM T30085 CLSY48 89630312 EC50 = 485 nM T30085 C6OGY1 89630313 EC50 = 598 nM T30085 CJXO12 89630320 EC50 = 151 nM T30085 CH64VU 89630321 EC50 = 315 nM T30085 CC8F3Z 89630327 EC50 = 649 nM T30085 C9YXG0 89630328 EC50 = 184 nM T30085 C3DYR9 89630335 EC50 = 335 nM T30085 CE90NZ 89630336 EC50 = 46 nM T30085 CB7D4P 89630337 EC50 = 678 nM T30085 CS7HD2 89630338 EC50 = 194 nM T30085 C54TXU 89630339 EC50 = 396 nM T30085 CS0JL9 89630340 EC50 = 1953 nM T30085 CQD86J 89630341 EC50 = 8541 nM T30085 CUA20I 89630342 EC50 = 431 nM T30085 COGX52 89630346 EC50 = 2251 nM T30085 CKQ8Z5 89630356 EC50 = 95 nM T30085 C7Y1CH 89634041 EC50 = 151 nM T30085 CR4IQ0 89634064 EC50 = 586 nM T30085 C68EIV 89634067 EC50 = 286 nM T30085 C5BX7V 89634086 EC50 = 655 nM T30085 CX98BP 89634088 EC50 = 429 nM T30085 C87NRT 89634090 EC50 = 2367 nM T30085 C9OL8G 89634110 EC50 = 2091 nM T30085 CCI4Y3 89634111 EC50 = 119 nM T30085 CI79TO 89634113 EC50 = 515 nM T30085 C0SP5V 89634117 EC50 = 2723 nM T30085 CIM9A6 89634124 EC50 = 211 nM T30085 CX82JF 90177831 IC50 = 14.5 nM T30085 CNZ3M2 90183119 IC50 = 3.7 nM T30085 C83KZC 90183140 IC50 = 1.6 nM T30085 C36FVE 90183231 IC50 = 3.7 nM T30085 C8L0ZD 90644321 IC50 = 5478 nM T30085 CJAW70 90644322 IC50 = 5699 nM T30085 CJR19O 90644323 IC50 = 9916 nM T30085 CZ09VO 90644324 IC50 = 9000 nM T30085 CJ9R8U 90644325 IC50 = 3296 nM T30085 C3OB6A 117642291 IC50 = 3.7 nM T30085 C37LUJ 127032843 EC50 = 1004 nM T30085 CO4ZI9 127033993 EC50 = 118 nM T30085 CUF5W6 127034238 EC50 = 284 nM T30085 C1QJ6A 127034239 EC50 = 249 nM T30085 CRGX75 127034242 EC50 = 588 nM T30085 C2M4ZJ 127034247 EC50 = 2591 nM T30085 C7JQ6C 129237363 IC50 = 22700 nM T30085 C8EN9I 133081837 IC50 = 2.5 nM T30085 CG36NB 133081841 IC50 = 2.5 nM T30085 CE26QS 133081845 IC50 = 2.5 nM T30085 CMI40H 133081848 IC50 = 3.4 nM T30085 CQC09F 133081850 IC50 = 3.1 nM T30085 C3ZMR2 133081853 IC50 = 1.3 nM T30085 CVB8A7 134469343 IC50 > 100 nM T30085 C95PDI 134469373 IC50 = 51.5 nM T30085 C5DF3L 134469421 IC50 = 47.2 nM T30085 CIB5Y9 134469475 IC50 = 42.4 nM T30085 CTN7F9 134469574 IC50 = 67.5 nM T30085 C81HPB 134469603 IC50 = 26.2 nM T30085 CDH70Y 134469622 IC50 = 69.4 nM T30085 C2HV3Z 134469646 IC50 = 51.3 nM T30085 C9U6KQ 134498364 IC50 = 1 nM T30085 C23TUN 134498374 IC50 = 1 nM T30085 C9C4XT 134498382 IC50 = 1 nM T30085 CX7R1U 134498384 IC50 = 3 nM T30085 CW4PQ9 134498385 IC50 = 1 nM T30085 CA2CX7 134498386 IC50 = 1 nM T30085 CX2V6Z 134498389 IC50 = 1 nM T30085 C1N6ZV 134498411 IC50 = 5 nM T30085 CA6TY7 134498420 IC50 = 1 nM T30085 CS3B7E 134498427 IC50 = 3 nM T30085 CC89KP 134498441 IC50 = 6 nM T30085 CD1F3O 134498886 IC50 = 2 nM T30085 C68VKL 134498938 IC50 = 3 nM T30085 C5M9BA 134498971 IC50 = 3 nM T30085 C8SWJ0 134499046 IC50 = 1 nM T30085 C41NYJ 134499051 IC50 = 10 nM T30085 C2DS4E 134512337 IC50 = 1 nM T30085 C6PO4L 135360405 IC50 = 42.3 nM T30085 CR7NU8 135360408 IC50 > 100 nM T30085 CVZ24G 135360416 IC50 > 100 nM T30085 CSV71C 135360417 IC50 > 100 nM T30085 C29PKS 135360449 IC50 > 100 nM T30085 CLK6D0 135360457 IC50 = 24 nM T30085 CZB1S9 135360458 IC50 = 63.5 nM T30085 CEY50H 135360459 IC50 > 100 nM T30085 CDL6A2 135360465 IC50 > 100 nM T30085 CU3ZF9 135360466 IC50 > 100 nM T30085 C2F8MH 135360468 IC50 > 100 nM T30085 C6G7YZ 135360474 IC50 > 100 nM T30085 COQP32 135360477 IC50 > 100 nM T30085 CK8DB1 135360478 IC50 = 15.9 nM T30085 CNZ5F6 135360652 IC50 > 100 nM T30085 CL9D0C 135360653 IC50 > 100 nM T30085 CZ6Q2E 135360662 IC50 = 29.7 nM T30085 C7R8AU 135360672 IC50 > 100 nM T30085 C7PHK5 135360761 IC50 > 100 nM T30085 C3BN6R 135360764 IC50 = 8.5 nM T30085 CD90SA 135360772 IC50 = 4.5 nM T30085 CGI31J 136059718 Ki = 12.4 nM T30085 CG91HF 137498460 IC50 = 5.3 nM T30085 CI9N6P 137498470 IC50 = 9 nM T30085 CP7R6L 137498479 IC50 = 23.2 nM T30085 C13MYJ 137498490 IC50 = 2.6 nM T30085 CXSR57 137498494 IC50 = 8.3 nM T30085 CTK58A 137498501 IC50 = 13.6 nM T30085 C76OXI 137498531 IC50 = 3 nM T30085 C5AZW2 137498544 IC50 = 62.3 nM T30085 CC0R7B 137498561 IC50 = 36 nM T30085 C89URP 137498572 IC50 = 7.5 nM T30085 CBR3V7 137631975 IC50 = 16400 nM T30085 C1Z2EB 137632973 IC50 = 5.9 nM T30085 CAV87T 137634442 IC50 = 5.9 nM T30085 CB1H9S 137635111 IC50 = 18.2 nM T30085 CX4T8B 137637304 IC50 = 31 nM T30085 CW28XT 137638119 IC50 = 1.1 nM T30085 CUFC09 137638493 IC50 = 1 nM T30085 C8RQG4 137639691 IC50 = 28.4 nM T30085 CO03BT 137639897 IC50 = 21.7 nM T30085 CNFX93 137640414 IC50 = 16700 nM T30085 C3KRZ6 137640660 IC50 = 3.4 nM T30085 C7IDG1 137642168 IC50 = 5 nM T30085 C4R5MT 137647890 IC50 = 9.1 nM T30085 CIK2X9 137648654 IC50 = 10.8 nM T30085 C87NEV 137652303 IC50 = 13.9 nM T30085 CB9ZF1 137654716 IC50 = 22.3 nM T30085 CLB4A6 137655093 IC50 = 6.8 nM T30085 CJMB48 137655785 IC50 = 21.3 nM T30085 CS1B6D 137656036 IC50 = 2.5 nM T30085 C2ZA4G 137661404 IC50 = 22.7 nM T30085 CY4PQ1 137661495 IC50 = 5.9 nM T30085 CY92AB 137661679 IC50 = 26200 nM T30085 CU43VR 137661793 IC50 = 4.4 nM T30085 CDN3R4 140930589 IC50 > 100 nM T30085 CBNS65 140930597 IC50 = 8.8 nM T30085 C4C6ZU 145949458 EC50 = 395 nM T30085 CXSG96 145949708 EC50 = 208 nM T30085 CD9KB2 145955593 EC50 = 370 nM T30085 CCT6Z8 145958861 EC50 = 457 nM T30085 C9PDG4 145959943 EC50 = 301 nM T30085 C0QLW6 145960082 EC50 = 204 nM T30085 CRSF74 145960900 IC50 = 1.03 nM T30085 CLOY80 145961834 IC50 = 1.08 nM T30085 CEI86V 145962549 IC50 = 0.63 nM T30085 CG1O8D 145962804 IC50 = 12.17 nM T30085 C54MKE 145963259 IC50 = 0.81 nM T30085 C8RG3X 145974336 EC50 = 173 nM T30085 CQ9MJ6 145979226 IC50 = 3 nM T30085 C2XS9K 145980077 IC50 = 7 nM T30085 C2MC3U 145981567 IC50 = 9 nM T30085 CP96KA 145983611 IC50 = 183.9 nM T30085 CQ5JG2 145983720 IC50 = 125.7 nM T30085 C27EKA 145984945 IC50 = 246.3 nM T30085 C7QIM1 145986927 IC50 = 5 nM T30085 C0NIQ8 145989102 IC50 = 4 nM T30085 CUP18S 145992935 IC50 = 36 nM T30085 C7QD1G 155511498 IC50 = 281 nM T30085 C62GZS 155512672 IC50 = 69 nM T30085 C0Y6AF 155513930 IC50 = 17 nM T30085 CXS5V9 155519466 IC50 = 798 nM T30085 CPKH72 155521866 IC50 = 10 nM T30085 C0L3BR 155527667 IC50 = 2126 nM T30085 CW9E6G 155527919 IC50 = 19 nM T30085 C6QYU8 155534804 IC50 = 84 nM T30085 C4Z3YH 155555849 IC50 = 34 nM T30085 C8FX9U 155556004 EC50 = 36 nM T30085 CDB31T 155559931 IC50 = 200 nM T30085 C2L5VQ 155568482 IC50 = 354 nM T30085 C27KZO 44580562 IC50 = 2400 nM T30085 C0UC5R 44580599 IC50 = 286 nM T30085 D00HFT 46229075 IC50 = 500 nM T30085 D01DIQ 46229072 IC50 = 40000 nM T30085 D03AJS 10177526 Ki = 2.4 nM T30085 D05AZW 46229071 IC50 = 40000 nM T30085 D06WAL 6072 IC50 = 16.4 nM T30085 D0HD2G 4788 IC50 = 18300 nM T30085 D0I2FC 15837283 IC50 = 35000 nM T30085 D0L8OJ 45269680 IC50 = 2000 nM T30085 D0M8EH 45488072 IC50 = 6.5 nM T30085 D0VE0Q 72936 IC50 = 4100 nM T30085 D0X1TN 9824918 IC50 = 260 nM T77350 D00UVA 11556711 IC50 = 14 nM T77350 D0SH3I 387447 IC50 = 3.3 nM T77350 D0DP0J 92135659 IC50 = 3000 nM T77350 D0F9BT 25067547 IC50 = 10 nM T77350 D0VO0T 24800541 IC50 = 3 nM T77350 CTB7A1 853170 Ki = 7900 nM T77350 CS1P9Y 906456 IC50 = 1600 nM T77350 CL9NX1 6610292 IC50 > 3000 nM T77350 CB2FX9 7012853 IC50 = 220 nM T77350 CLU69K 10628969 IC50 = 630 nM T77350 CHIG24 12437395 Ki = 1800 nM T77350 CV5A0C 13494006 Ki = 2000 nM T77350 C4M3CI 25126032 IC50 = 22 nM T77350 CP78TJ 25127030 IC50 = 238 nM T77350 C8F0CI 25127659 IC50 = 41 nM T77350 CLT5F4 25128327 IC50 = 607 nM T77350 CT5ZA0 42638620 IC50 = 21 nM T77350 C9OG6U 42638621 IC50 = 5 nM T77350 C8TPJ6 42638622 IC50 = 36 nM T77350 CSR4Z3 42639306 IC50 = 93 nM T77350 CZNA09 44464211 Ki = 1100 nM T77350 C2VY4L 44464464 Ki = 3500 nM T77350 C06QXA 44464465 Ki = 1100 nM T77350 CB3M9F 44591653 IC50 = 784 nM T77350 CH67EX 44591654 IC50 = 82 nM T77350 CV1P6X 56945245 IC50 > 10000 nM T77350 CMPN64 71290695 Ki = 1400 nM T77350 C45HOE 71562349 IC50 = 1170 nM T77350 CGY43C 78425867 IC50 = 34 nM T77350 CWPX04 86288853 Ki = 3500 nM T77350 CBL1U6 89449895 IC50 = 13 nM T77350 CFPT98 90655054 IC50 = 31 nM T77350 C5JZ8R 90655055 IC50 = 59 nM T77350 CM7V1L 90655870 Ki = 520 nM T77350 CIY89A 90655872 Ki = 6000 nM T77350 CTHX07 90655873 Ki = 1200 nM T77350 CC0OF1 101874274 IC50 = 6.6 nM T77350 CG0N1O 101874275 IC50 = 8.3 nM T77350 CL50TR 101874276 IC50 = 36 nM T77350 C0RY3V 101874277 IC50 = 32 nM T77350 CVHC29 101874278 IC50 = 53 nM T77350 C4VHU6 101874279 IC50 = 11 nM T77350 C9C5OZ 117607839 IC50 = 23 nM T77350 C9BZ6E 117607841 IC50 = 29 nM T77350 CLHS74 117607901 IC50 = 83 nM T77350 CW9R0U 117607904 IC50 = 0.039 nM T77350 CKPU97 117607978 IC50 = 262 nM T77350 C7QST8 117611788 IC50 = 4274 nM T77350 C2QDO6 117611839 IC50 = 38 nM T77350 CO1HJ9 117611880 IC50 = 4810 nM T77350 CZ6C1M 117611892 IC50 = 3 nM T77350 C9YH1X 117611941 IC50 = 44639 nM T77350 C31HNL 117612022 IC50 = 5 nM T77350 C35YHK 118709573 IC50 > 50000 nM T77350 CWBF42 118709574 IC50 = 2 nM T77350 CLUS08 118709575 IC50 = 3.1 nM T77350 CUYG85 118709576 IC50 = 244 nM T77350 C3X5ZP 118709577 IC50 = 5 nM T77350 CZL52Y 118709661 IC50 = 3 nM T77350 C23GJD 118709662 IC50 = 14 nM T77350 C2J0CS 118709663 IC50 = 1.4 nM T77350 CV49FN 118709664 IC50 = 2.1 nM T77350 CC85SD 118709665 IC50 = 1.2 nM T77350 CBCF19 118709666 IC50 = 3.3 nM T77350 C29DIE 118709667 IC50 = 392 nM T77350 CAJ1Z2 118709668 IC50 = 5700 nM T77350 CC7FO9 118709669 IC50 = 632 nM T77350 C1DP4N 118899141 IC50 = 57 nM T77350 CUH45I 118899149 IC50 = 14 nM T77350 CA83ML 118899158 IC50 = 5.5 nM T77350 C0OLW2 122204528 IC50 = 681.1 nM T77350 C6C0JB 122576692 IC50 = 13 nM T77350 C3P0QD 122576697 IC50 = 9 nM T77350 CT96PH 129047769 IC50 = 169 nM T77350 CI24DQ 129047778 IC50 = 24 nM T77350 CI2J8F 129047830 IC50 = 4 nM T77350 C7BGS2 129047963 IC50 = 15 nM T77350 CC10QA 136498865 Ki = 1700 nM T77350 C1JH8K 138545006 IC50 > 100000 nM T77350 CLT78F 138545112 IC50 > 100000 nM T77350 C7DZ8K 138545235 IC50 > 100000 nM T77350 CIS28V 139209090 IC50 = 26 nM T77350 CB46AI 139209092 IC50 = 7890 nM T77350 CL45BO 145960456 IC50 > 100000 nM T77350 C5G6LM 145961320 IC50 = 3100 nM T77350 CUIF27 145961566 IC50 = 14000 nM T77350 CI9JH6 145961877 IC50 = 6700 nM T77350 C3M4OD 145961898 IC50 = 17200 nM T77350 C8CSZ0 145962247 IC50 = 136500 nM T77350 C97URS 145962850 IC50 = 450 nM T77350 COA19G 145963426 IC50 > 100000 nM T77350 C9BWP4 145979302 IC50 = 10000 nM T77350 CN79HG 145979487 IC50 = 2700 nM T77350 CEI3U1 145979850 IC50 = 5200 nM T77350 CG6UL0 145980995 IC50 = 2700 nM T77350 CB67YT 145981691 IC50 = 1600 nM T77350 C41IRV 145981707 IC50 = 260 nM T77350 CL1F8N 145982922 IC50 = 19700 nM T77350 C5X3GQ 145986425 IC50 = 7800 nM T77350 CRZE86 145986857 IC50 = 3960 nM T77350 CHWT73 145987085 IC50 = 6100 nM T77350 CM3H4F 145987197 IC50 = 3800 nM T77350 CNZ7R6 145987536 IC50 = 13200 nM T77350 C1EF3B 145988020 IC50 = 10.2 nM T77350 CQIS01 145988427 IC50 = 6500 nM T77350 C4R3HC 145988596 IC50 = 18.6 nM T77350 CN8K1E 145989337 IC50 = 9.1 nM T77350 CE16JH 145989568 IC50 = 170 nM T77350 CXG30R 145990249 IC50 = 12600 nM T77350 CWS03B 145991519 IC50 = 41.2 nM T77350 C8G1BT 145991875 IC50 = 17100 nM T77350 C8IL9E 145992200 IC50 = 3930 nM T77350 C9OHR3 145992219 IC50 = 44.7 nM T77350 CBY18W 145992498 IC50 = 1900 nM T77350 CCU34H 145992780 IC50 = 420 nM T77350 C6GHQ9 145993211 IC50 = 25100 nM T77350 CEVY70 145993649 IC50 = 572 nM T77350 CJO08K 145993925 IC50 = 200 nM T77350 C0T3WE 155510481 IC50 = 351 nM T77350 CVA50J 155512274 IC50 = 141 nM T77350 C8E6ZX 155514792 IC50 = 2200 nM T77350 C0SDO2 155515259 IC50 > 10000 nM T77350 CX76LO 155515463 IC50 = 19 nM T77350 CSD4T9 155515790 IC50 = 1010 nM T77350 C53ZEN 155516179 IC50 > 10000 nM T77350 CM3BV8 155516620 IC50 > 100000 nM T77350 C4VT1Y 155517101 IC50 = 112 nM T77350 CE95IQ 155518158 IC50 > 100000 nM T77350 CFQZ35 155518266 IC50 = 100 nM T77350 CEF5D1 155519196 IC50 = 3111 nM T77350 CEJ56T 155519405 IC50 = 179 nM T77350 CNM0Q9 155521286 IC50 > 10000 nM T77350 CZKF54 155521690 IC50 = 2800 nM T77350 C8NOH2 155521815 IC50 = 195 nM T77350 C8GNQ9 155522828 IC50 = 346 nM T77350 CW75YK 155523151 IC50 > 100000 nM T77350 C78BVM 155526764 IC50 = 24 nM T77350 CAC34Y 155527225 IC50 = 4100 nM T77350 CPHX68 155527880 IC50 = 32 nM T77350 C3PMD9 155529033 IC50 = 38 nM T77350 C6GQR9 155531009 IC50 = 120 nM T77350 CUP2B4 155531358 IC50 = 49 nM T77350 CD84AS 155531896 IC50 = 4690 nM T77350 CEF08Q 155534115 IC50 = 9970 nM T77350 CT35RL 155534506 IC50 = 226 nM T77350 COZ5V6 155535430 IC50 = 2350 nM T77350 CJY7W1 155535900 IC50 = 227 nM T77350 CCYI81 155537845 IC50 = 2090 nM T77350 C2NTI6 155538936 IC50 = 28400 nM T77350 C6E1YP 155539344 IC50 > 100000 nM T77350 CX3HR1 155540804 IC50 = 200 nM T77350 CT2V8E 155540850 IC50 = 475 nM T77350 CQE43H 155541095 IC50 = 20100 nM T77350 C13VXP 155541111 IC50 = 264 nM T77350 C6OIY3 155541618 IC50 > 100000 nM T77350 C41IBR 155542489 IC50 = 128 nM T77350 C6GIE2 155546910 IC50 = 174 nM T77350 CKY05M 155547055 IC50 = 763 nM T77350 CA8Z7D 155548324 IC50 = 200 nM T77350 C8HVD1 155548349 IC50 = 3560 nM T77350 CIM5K2 155549227 IC50 = 6340 nM T77350 C12LPX 155551071 IC50 = 35 nM T77350 CBHM14 155553205 IC50 > 100000 nM T77350 C35NJC 155553210 IC50 > 10000 nM T77350 CI15FC 155553565 IC50 > 10000 nM T77350 CVJ3E7 155553910 IC50 = 46 nM T77350 C12WHV 155553963 IC50 = 1830 nM T77350 C6YP0L 155554916 IC50 > 100000 nM T77350 CP58EH 155556856 IC50 = 1400 nM T77350 CCLI81 155557971 IC50 = 433 nM T77350 C0Z4ET 155558668 IC50 = 72.7 nM T77350 CMH7V5 155559237 IC50 = 2090 nM T77350 CZ3XY4 155563335 IC50 = 5650 nM T77350 CV9C2Z 155564821 IC50 = 365 nM T77350 C3N8XZ 155564979 IC50 = 384 nM T77350 CEAV80 155566012 IC50 = 38 nM T77350 CU53FD 155566562 IC50 > 10000 nM T77350 C5Z7YC 155567712 IC50 = 2100 nM T77350 CG2KN0 155567727 IC50 = 2892 nM T77350 CV68GZ 155568757 IC50 = 13 nM T77350 C4ZV3Q 155568941 IC50 > 10000 nM T77350 D0K7CX 325597 Ki = 420 nM T77350 D0Q4MO 23642227 IC50 = 18 nM T15888 CZN6S9 743974 EC50 > 25118.86 nM T15888 C6ENV5 100951623 IC50 > 10000 nM T15888 C5AX9S 155516007 IC50 = 8400 nM T15888 CC3H4U 155518713 EC50 = 5200 nM T15888 C4H2DQ 155519352 IC50 = 38 nM T15888 C2LS4J 155519637 EC50 = 2300 nM T15888 CR35QE 155519969 IC50 = 1200 nM T15888 CNP0X5 155520796 IC50 > 3000 nM T15888 C4YWV9 155525712 IC50 = 7600 nM T15888 C3HGV5 155526368 IC50 = 2800 nM T15888 C3BV0S 155530073 EC50 = 2700 nM T15888 CHE2I9 155531953 IC50 = 110 nM T15888 C8HM6F 155535518 IC50 = 940 nM T15888 CDB2A4 155535988 IC50 = 32 nM T15888 C05UQJ 155537257 EC50 = 3900 nM T15888 CW1F7Y 155538284 IC50 = 3300 nM T15888 C43DZF 155538662 EC50 = 1500 nM T15888 CG6VC8 155543662 IC50 = 2400 nM T15888 CFR62J 155544237 IC50 = 37 nM T15888 C2PE7M 155546659 EC50 > 10000 nM T15888 C3M2QO 155548932 EC50 = 3900 nM T15888 C0XEJ7 155550204 IC50 = 3400 nM T15888 CW4D3J 155550367 IC50 = 3300 nM T15888 CU5XR3 155554813 EC50 > 10000 nM T15888 C2THI9 155554828 EC50 = 940 nM T15888 CDT78C 155558601 EC50 > 3000 nM T15888 CN3U1L 155561023 EC50 > 10000 nM T15888 C0YOS1 155563693 EC50 = 1300 nM T15888 C3EKH7 155564611 IC50 = 4300 nM T15888 C6OES3 155567133 IC50 = 2500 nM T15888 CMG5R7 155569501 EC50 = 8300 nM T71081 D0W4HZ 148195 IC50 = 70 nM T71081 CF4V6K 513439 IC50 = 8000 nM T71081 CN5FE6 513441 IC50 > 300000 nM T71081 CK5H4S 9810043 IC50 = 14300 nM T71081 CQ8WP7 9833296 IC50 = 180 nM T71081 C5C2NJ 9939360 IC50 = 4300 nM T71081 CT8P7B 9939571 IC50 = 5000 nM T71081 CLVD03 9940233 IC50 = 20 nM T71081 C9ZB2I 10055858 IC50 = 20 nM T71081 CY1DC9 10100867 IC50 = 310 nM T71081 CGDL43 10508557 IC50 = 6300 nM T71081 CW84BC 10556304 IC50 = 570 nM T71081 CAR49J 10699791 IC50 > 1000 nM T71081 CSR0T2 10746913 IC50 = 300 nM T71081 C1HBJ0 10770859 IC50 = 88 nM T71081 CCAI68 10771001 IC50 > 1000 nM T71081 CIW4F5 10794573 IC50 = 180 nM T71081 CI26KD 10818103 IC50 = 710 nM T71081 C3V7SW 10818236 IC50 = 400 nM T71081 CV5XQ4 11802593 IC50 = 190 nM T71081 CW10OJ 11802840 IC50 = 330 nM T71081 C9EAM6 12083952 IC50 = 15 nM T71081 CV21AS 44302820 IC50 = 16000 nM T71081 C65XOW 44302991 IC50 = 14000 nM T71081 C75JNV 44302992 IC50 = 12000 nM T71081 CIKL28 44303071 IC50 = 1500 nM T71081 CY4K2N 44303176 IC50 = 10000 nM T71081 C1N0QO 44303225 IC50 = 10000 nM T71081 C3TR6P 44303262 IC50 = 80000 nM T71081 C3R9GO 44303277 IC50 = 15000 nM T71081 C9VSH1 44303334 IC50 = 50000 nM T71081 C12YJD 44303350 IC50 = 6700 nM T71081 CX6EL9 44303355 IC50 = 1000 nM T71081 CD5KC7 44303358 IC50 = 10500 nM T71081 CBDJ05 44303385 IC50 = 8000 nM T71081 C23FEC 44303394 IC50 = 14000 nM T71081 C0RO6G 44303429 IC50 = 27000 nM T71081 CL4RM9 44323680 IC50 = 15 nM T71081 C75QIV 44323695 IC50 = 15 nM T71081 CN2JH6 44323892 IC50 = 15 nM T71081 CS3CD6 44333466 IC50 > 200000 nM T71081 C0ZUC8 44386438 IC50 = 35000 nM T71081 C0M6NS 44559702 IC50 = 2 ug.mL-1 T71081 CSQ89F 82709780 IC50 = 320000 nM T71081 CVA6E2 90665525 IC50 = 80000 nM T71081 C20-OCT 90665526 IC50 = 80000 nM T71081 C8VM1S 90665527 IC50 = 100000 nM T71081 D0BS6Q 3115 IC50 = 200 nM T11453 C41AIU 11169089 IC50 = 2000 nM T11453 CU4J6H 11249762 IC50 = 3200 nM T11453 COE04Q 11352811 IC50 > 10000 nM T11453 CG43XJ 11376210 IC50 = 4900 nM T11453 C8J4UT 11410779 IC50 = 1000 nM T11453 CP56DO 11599295 IC50 = 6000 nM T11453 C5B9GH 44561391 IC50 > 1000 nM T11453 C6F4EX 44561438 IC50 = 2500 nM T11453 CSB74O 44561439 IC50 = 2800 nM T11453 C5A8MI 44561440 IC50 > 1000 nM T11453 CQU45G 44561479 IC50 > 1000 nM T11453 CE4N0X 44561480 IC50 > 1000 nM T11453 C9Y2NP 44561556 IC50 = 3000 nM T59881 D08FJL 16681432 EC50 = 4.8 nM T59881 D0D8XY 5311010 Ki = 44 nM T59881 D0M3FJ 439302 EC50 = 0.2 nM T59881 D0N4OW 644077 EC50 = 0.0035 nM T59881 D0U7SH 5311065 Ki = 5.8 nM T59881 D04QZI 11340891 Ki > 10000 nM T59881 D09WYL 11634973 Ki > 7943.28 nM T59881 D0S3YN 53330936 EC50 = 338.84 nM T59881 D0SY9B 9895468 Ki = 0.6 nM T59881 D03RYS 5311500 Ki > 1000 nM T59881 D0A1KU 11683187 Ki > 10000 nM T59881 D0AV0O 3038506 IC50 > 100000 nM T59881 C0R7SI 449224 EC50 = 180 nM T59881 C5F1ST 1103817 Ki > 10000 nM T59881 CO3SD6 9811830 EC50 = 25 nM T59881 CR6VX2 10483105 Ki = 1300 nM T59881 C0FJM7 11194023 Ki = 12.8 nM T59881 CO3A5Z 11240155 Ki = 3.4 nM T59881 CC0KT1 11251777 Ki = 14.8 nM T59881 CUED54 11257380 Ki > 10000 nM T59881 C5OTG4 11274745 Ki = 156 nM T59881 C9T8BV 11286254 Ki = 7.8 nM T59881 CB6TF8 11297732 Ki = 9.5 nM T59881 CPND10 11389106 Ki = 2 nM T59881 CEM1X7 11400547 Ki = 0.52 nM T59881 CR4N5I 11465834 Ki < 6309.57 nM T59881 CM83DS 11468862 Ki = 1.8 nM T59881 COC7Q9 11488952 Ki < 6309.57 nM T59881 CQ96XZ 11569194 Ki < 6309.57 nM T59881 C60DKW 11569672 Ki < 50118.72 nM T59881 CG7CL9 11578939 EC50 = 44 nM T59881 CY0HE4 11677610 IC50 = 3 nM T59881 C91CIO 11815584 Ki = 1.5 nM T59881 C8GC2P 11854507 IC50 = 6 nM T59881 C5A9MK 11854509 IC50 = 7 nM T59881 C14VXM 11854759 IC50 = 9 nM T59881 C4CTD2 14257660 EC50 = 7.5 nM T59881 CHU5E4 16051933 Ki = 0.37 nM T59881 CG6T2S 24900844 IC50 = 1 nM T59881 CDO2Q8 25059334 Ki = 5 nM T59881 COC73W 25212177 Ki = 31.62 nM T59881 CY67HA 42611262 Ki = 1258.93 nM T59881 CB82ZC 44232512 EC50 = 450 nM T59881 CBV47F 44243143 Ki > 10000 nM T59881 CDI2Q4 44247566 IC50 = 15.85 nM T59881 CVI6Q3 44275104 Ki = 5.9 nM T59881 CW7JM3 44275447 Ki = 9.4 nM T59881 C2J8GK 44316235 Ki = 6.5 nM T59881 CIE6Y1 44316236 Ki = 22.9 nM T59881 C24NQS 44316241 Ki = 0.23 nM T59881 CYBF69 44465987 IC50 = 316.23 nM T59881 CB17SO 44465990 IC50 = 1000 nM T59881 CB1A5H 44466236 IC50 = 5.012 nM T59881 CLE7W0 44466239 IC50 = 3.981 nM T59881 CU6XQ1 44466493 IC50 = 158.49 nM T59881 CPA4W5 44467270 IC50 = 12.59 nM T59881 CKA3S0 44467347 IC50 = 10 nM T59881 C2LF9D 44467348 IC50 = 2.512 nM T59881 CMYW04 44467349 IC50 = 63.1 nM T59881 CC1AY9 44467496 IC50 = 794.33 nM T59881 CMD57H 44467497 IC50 = 79.43 nM T59881 COJI26 44467563 IC50 = 251.19 nM T59881 CJHN89 44467564 IC50 = 63.1 nM T59881 CVFO29 44467565 IC50 = 12.59 nM T59881 CK7YC4 44467566 IC50 = 50.12 nM T59881 CCS6Z5 44467632 IC50 = 6.31 nM T59881 CTS2X3 44467634 IC50 = 501.19 nM T59881 CY57ZB 44467635 IC50 = 79.43 nM T59881 CYMW64 44467636 IC50 = 794.33 nM T59881 C89XHW 44467698 IC50 = 1258.93 nM T59881 CG2DZ6 44467699 IC50 = 630.96 nM T59881 CB9I3Q 44467700 IC50 = 125.89 nM T59881 CAQ63W 44467701 IC50 = 199.53 nM T59881 CW2YN9 44467702 IC50 = 3981.07 nM T59881 CUT45Y 44467771 IC50 = 5.012 nM T59881 CY98GZ 44467773 IC50 = 63.1 nM T59881 CYK02B 44467774 IC50 = 630.96 nM T59881 CNZ23K 44467775 IC50 = 3.981 nM T59881 CNF41X 44467845 IC50 = 1258.93 nM T59881 C3JC8N 44467846 IC50 = 501.19 nM T59881 CK97TD 44467847 IC50 = 1258.93 nM T59881 CL8CP7 44467848 IC50 = 1258.93 nM T59881 C93APB 44467913 IC50 = 501.19 nM T59881 CH4Y6E 44467914 IC50 = 63.1 nM T59881 C3S8KD 44467916 IC50 = 6.31 nM T59881 C87BTI 44467917 IC50 = 199.53 nM T59881 C7FWI5 44467978 IC50 = 398.11 nM T59881 C9F4QJ 44467979 IC50 = 5.012 nM T59881 C8MC9S 44467981 IC50 = 199.53 nM T59881 CWIB10 44467982 IC50 = 5.012 nM T59881 C9SY5P 44468051 IC50 = 100 nM T59881 C6C8ST 44468052 IC50 = 63.1 nM T59881 CDN81V 44468053 IC50 = 199.53 nM T59881 CZ16PM 44468115 IC50 = 6.31 nM T59881 CX82BQ 44468117 IC50 = 10 nM T59881 CKY0U5 44468118 IC50 = 63.1 nM T59881 CLCK14 44579399 Ki > 10000 nM T59881 C5OSG6 45483182 Ki = 1137 nM T59881 CZBU35 45483183 Ki = 1036 nM T59881 C8GVN6 45483194 Ki = 416 nM T59881 C6I9KO 45483202 Ki = 413 nM T59881 CQ3BL0 45483203 Ki = 138 nM T59881 CYQ36K 45483204 Ki = 43.65 nM T59881 CYX27Z 45483235 Ki = 295 nM T59881 CEIU28 45483236 Ki = 66 nM T59881 C06EOV 45483237 Ki = 96 nM T59881 CUJ8V3 45483238 Ki = 104 nM T59881 C4TZ6D 45483239 Ki = 218 nM T59881 CT9B5J 45483240 Ki = 939 nM T59881 C45UJI 45483241 Ki = 279 nM T59881 C75VPW 45483242 Ki = 717 nM T59881 C7IED0 45483243 Ki = 122 nM T59881 CE5M9W 45483247 Ki = 7196 nM T59881 CY95GV 45483255 Ki = 600 nM T59881 CWA23E 45483256 Ki = 152 nM T59881 C4ANR9 45483282 Ki = 1184 nM T59881 CJM89E 45483300 Ki = 114 nM T59881 CYA3F4 45483320 Ki = 1523 nM T59881 CPYH25 45483321 Ki = 715 nM T59881 C6CI2W 45483323 Ki = 748 nM T59881 C02MEC 45483324 Ki = 35 nM T59881 CH73EJ 45483325 Ki = 78 nM T59881 C14SKI 46934433 IC50 = 310 nM T59881 CUWG39 46934434 IC50 = 120 nM T59881 C4XZ5I 49865463 IC50 = 15.85 nM T59881 CR3UF5 49865507 IC50 = 398.11 nM T59881 CX6L0Q 49865609 IC50 > 100000 nM T59881 CIF6O3 49865610 IC50 = 22000 nM T59881 C68RMB 49865611 IC50 = 1700 nM T59881 CCOM93 49865612 IC50 = 4800 nM T59881 C2TX8J 49865645 IC50 = 25800 nM T59881 CRWT29 49865646 IC50 = 7600 nM T59881 CN6K4P 49865647 IC50 = 3800 nM T59881 CXCF32 49865670 IC50 = 1800 nM T59881 CZDG69 49865671 IC50 = 340 nM T59881 C1X6IO 49865672 IC50 = 710 nM T59881 CT2O0N 49865673 IC50 = 1100 nM T59881 C5W0IM 49866180 IC50 = 200 nM T59881 CPJ5K8 49866181 IC50 = 5100 nM T59881 CLV51T 49866220 IC50 = 30500 nM T59881 C6A1VE 49866221 IC50 > 100000 nM T59881 C7QU6V 49866222 IC50 > 100000 nM T59881 C73UEW 49866223 IC50 = 2100 nM T59881 C9VE1B 49866245 IC50 = 4000 nM T59881 C8GK6S 49866246 IC50 = 3600 nM T59881 C2V4GY 49866247 IC50 > 30000 nM T59881 CK08EY 49866248 IC50 > 30000 nM T59881 C48PQT 50915110 Ki = 125.89 nM T59881 CO4WH0 50941635 Ki = 158.49 nM T59881 CMPE57 52941704 Ki = 208 nM T59881 CBDS48 52949017 Ki = 44 nM T59881 C0KBC6 53316694 Ki = 25.12 nM T59881 CQ43EC 53316695 Ki = 100 nM T59881 CWXA96 53316696 Ki = 501.19 nM T59881 C9N1GY 53316697 Ki = 630.96 nM T59881 CI4E7O 53316698 Ki = 398.11 nM T59881 C5Z7NE 53316699 Ki = 794.33 nM T59881 C8EBM3 53316700 Ki = 1995.26 nM T59881 C4M0LW 53316701 Ki = 251.19 nM T59881 CUL83M 53316870 IC50 = 366 nM T59881 CLWX14 53316871 IC50 = 125 nM T59881 C8NSI3 53316944 IC50 = 6050 nM T59881 C6Q5XO 53316945 IC50 = 4 nM T59881 CUNZ51 53316999 IC50 = 2500 nM T59881 C9YP1M 53317000 IC50 = 46 nM T59881 CH47QY 53317994 Ki = 100 nM T59881 CYF57C 53317995 Ki = 1258.93 nM T59881 CQB5U6 53317996 Ki = 398.11 nM T59881 CYKN31 53317997 Ki = 630.96 nM T59881 C45YNR 53318240 IC50 = 644 nM T59881 CIA5M3 53318279 IC50 > 20000 nM T59881 CH1XY8 53318916 IC50 = 5 nM T59881 CZ6IN4 53319343 Ki = 158.49 nM T59881 CBV9Z5 53319602 IC50 = 328 nM T59881 CBS5V0 53319603 IC50 = 86 nM T59881 CP7Q8L 53319604 IC50 = 122 nM T59881 CHIU02 53319605 IC50 > 20000 nM T59881 C42OPZ 53320648 Ki = 316.23 nM T59881 C2WET7 53320829 IC50 = 1030 nM T59881 C1HB2P 53320890 IC50 = 1350 nM T59881 C1V4OY 53320891 IC50 = 59 nM T59881 CL7IK0 53320892 IC50 > 20000 nM T59881 CN7Z4W 53320940 IC50 > 20000 nM T59881 CSTR80 53321851 Ki = 398.11 nM T59881 CW0CP5 53321939 Ki = 100 nM T59881 CIP52X 53321940 Ki = 3162.28 nM T59881 CI15MR 53322162 IC50 = 1450 nM T59881 CTDW75 53322163 IC50 = 800 nM T59881 C4E1XF 53322164 IC50 = 30 nM T59881 C5NBE4 53322230 IC50 = 470 nM T59881 C2UM3L 53322231 IC50 = 2400 nM T59881 CXJ4C2 53322269 IC50 = 152 nM T59881 CP3A9G 53322270 IC50 = 17 nM T59881 CCE69T 53322990 IC50 = 34 nM T59881 CS0Q9A 53323297 Ki = 100 nM T59881 CLK0X6 53323298 Ki = 316.23 nM T59881 C7K5ID 53323615 IC50 = 2350 nM T59881 CVK3H4 53323616 IC50 = 72 nM T59881 CS2XJ4 53323617 IC50 = 49 nM T59881 CLK3Q1 53324234 IC50 = 250 nM T59881 C1X2ND 53324324 Ki = 1258.93 nM T59881 CVB45I 53324622 Ki = 2511.89 nM T59881 CZO92E 53324623 Ki = 1000 nM T59881 C1ASK4 53324624 Ki = 501.19 nM T59881 CE2G1A 53324625 Ki = 1258.93 nM T59881 CDV2M3 53324811 IC50 = 113 nM T59881 COQ4U2 53324871 IC50 = 3100 nM T59881 CTQX04 53324872 IC50 = 325 nM T59881 CK4J6G 53324873 IC50 = 26 nM T59881 C7B6LE 53325559 IC50 = 42 nM T59881 C24KRL 53325929 Ki = 398.11 nM T59881 C91IME 53325930 Ki = 794.33 nM T59881 CSMW36 53325931 Ki = 1258.93 nM T59881 C0I2DT 53325932 Ki = 630.96 nM T59881 CG73VQ 53325933 Ki = 1258.93 nM T59881 CG8JN6 53326089 IC50 = 15 nM T59881 CYLU08 53326194 IC50 = 196 nM T59881 C4TEY2 53358902 Ki = 190 nM T59881 C5FA7N 53358903 Ki = 180 nM T59881 CRSC15 53358904 Ki = 63 nM T59881 C63IVJ 53362154 EC50 = 147.91 nM T59881 C21HMW 53362155 EC50 = 28 nM T59881 CF60LM 53362156 EC50 = 537.03 nM T59881 CGMY47 53362202 EC50 = 70 nM T59881 C9V8RI 53362203 EC50 = 28.84 nM T59881 CAL1Y3 53362204 EC50 = 38.9 nM T59881 C6N5EX 53362257 EC50 = 29.51 nM T59881 CS40QD 53362258 EC50 = 62 nM T59881 CFWL28 53362259 EC50 = 56 nM T59881 CNDR76 53362310 EC50 = 25.7 nM T59881 COUH09 53362311 EC50 = 19 nM T59881 C1MU4B 53362312 EC50 = 61.66 nM T59881 CLRT87 53362368 EC50 = 27.54 nM T59881 CG8J6H 53362369 EC50 = 41 nM T59881 CD1N3U 53362370 EC50 = 45.71 nM T59881 CRY95P 53362428 EC50 = 208.93 nM T59881 C3TFA8 53362429 EC50 = 74 nM T59881 C4U1PT 53362430 EC50 = 38 nM T59881 C09KLV 53362488 EC50 = 31.62 nM T59881 CRX54F 53362489 EC50 = 100 nM T59881 C3KCI9 53362490 EC50 = 954.99 nM T59881 CW32MV 53362546 EC50 = 37 nM T59881 C5EG6T 53362547 EC50 = 8.7 nM T59881 CUD9F0 53362548 EC50 = 20.89 nM T59881 CVJ9U2 53362603 EC50 = 250 nM T59881 CMY7V4 53362604 EC50 = 64.57 nM T59881 CK9V1G 53362605 EC50 = 117.49 nM T59881 CCRZ83 53362670 EC50 = 30.9 nM T59881 CYK9B3 53362671 EC50 = 570 nM T59881 CCK0P6 53362672 EC50 = 524.81 nM T59881 CYG85M 53362729 EC50 = 26 nM T59881 C1IBT7 53362730 EC50 = 1778.28 nM T59881 CI0F3Y 53362731 EC50 = 457.09 nM T59881 C3XW1F 53362732 EC50 = 220 nM T59881 CYTJ92 53362793 EC50 > 10000 nM T59881 CQ9CD8 53362794 EC50 = 194.98 nM T59881 CAN2C1 53362795 EC50 = 360 nM T59881 CO4UA0 53362796 EC50 = 363.08 nM T59881 C0NSZ5 53362797 EC50 = 510 nM T59881 CFJO73 53362798 EC50 = 260 nM T59881 C2RSW6 53362849 EC50 = 430 nM T59881 C5K9YV 53362850 EC50 = 150 nM T59881 CB3AR7 53362851 EC50 = 50 nM T59881 C42SJF 53362852 EC50 = 346.74 nM T59881 C8U6LX 53362853 EC50 = 380 nM T59881 CH93SM 53362854 EC50 = 104.71 nM T59881 C7RYJ0 53362909 EC50 = 208.93 nM T59881 CKV9D6 53362910 EC50 > 10000 nM T59881 CX9YM6 53362911 EC50 = 43.65 nM T59881 C76TQB 53362913 EC50 = 117.49 nM T59881 C5XCD8 53362914 EC50 = 120 nM T59881 C8N0TX 53362915 EC50 = 75.86 nM T59881 CU9X3P 53362962 EC50 = 250 nM T59881 C61CNE 53362963 EC50 = 19.5 nM T59881 CF30CI 53362964 EC50 = 7.943 nM T59881 C6SB7W 53362965 EC50 = 109.65 nM T59881 C32FZM 53362966 EC50 = 140 nM T59881 CJ06TA 53362967 EC50 = 17.78 nM T59881 C6AN7Y 53363015 EC50 = 63.1 nM T59881 C52IOF 53363016 EC50 = 58.88 nM T59881 C1SHU3 53363017 EC50 = 97 nM T59881 CNA2L1 53364234 Ki > 10000 nM T59881 C3L7RP 54580516 Ki = 0.03 nM T59881 C16GUQ 54580517 Ki > 10000 nM T59881 CX1H3Z 54580518 Ki = 1.3 nM T59881 C9S8KL 54580830 IC50 = 275 nM T59881 C5A1IH 54580831 IC50 = 397 nM T59881 CB40UM 54580832 IC50 = 9 nM T59881 CK5BC6 54580862 Ki > 10000 nM T59881 CTV6R8 54580863 Ki = 500 nM T59881 CP0FE9 54580874 Ki = 250 nM T59881 C7X4LI 54581307 Ki = 1.3 nM T59881 CB5R2M 54581528 Ki = 3.8 nM T59881 CR7GD2 54581529 Ki = 0.26 nM T59881 CUW8C7 54581530 Ki = 0.03 nM T59881 C0V5XG 54581531 Ki = 786 nM T59881 CJM92I 54581532 Ki = 276 nM T59881 CD21EL 54581533 Ki = 2 nM T59881 CAR8F0 54581876 IC50 > 20000 nM T59881 CW2E5R 54581877 IC50 = 642 nM T59881 CS7FZ5 54581878 IC50 = 2350 nM T59881 C7NGK4 54581879 IC50 = 19 nM T59881 CE39JS 54581880 IC50 = 610 nM T59881 CTG89K 54581898 IC50 = 37 nM T59881 CY82GR 54581930 Ki = 10000 nM T59881 C0ZNY9 54582318 Ki = 3.7 nM T59881 CQ7Z8U 54582526 Ki = 3.9 nM T59881 C49HXA 54582805 IC50 = 79 nM T59881 CK4VJ9 54582806 IC50 = 320 nM T59881 C0B1QP 54582807 IC50 = 46 nM T59881 CM34LD 54582808 IC50 = 77 nM T59881 CX81DP 54582817 IC50 = 700 nM T59881 CLAE74 54582843 Ki = 630 nM T59881 C27LJC 54582853 Ki = 2500 nM T59881 C4F2XW 54583496 Ki = 101 nM T59881 CF2UP6 54583578 Ki = 1200 nM T59881 C37RSZ 54583807 IC50 = 388 nM T59881 CM9B8I 54583808 IC50 = 238 nM T59881 CP6B4S 54583859 Ki = 500 nM T59881 CTH30C 54583860 Ki = 310 nM T59881 C5NV8X 54583861 Ki = 260 nM T59881 C9YV3Q 54584201 Ki = 1258.93 nM T59881 C7MP0S 54584254 Ki >= 10000 nM T59881 C73IGF 54584265 Ki = 0.52 nM T59881 CX5T1G 54584266 Ki = 0.65 nM T59881 CIGN05 54584267 Ki = 0.61 nM T59881 CC49GD 54584268 Ki = 8.4 nM T59881 C9N2QH 54584476 Ki = 1.3 nM T59881 CD1A0H 54584477 Ki = 26 nM T59881 CXPY04 54584478 Ki = 0.08 nM T59881 CV32SD 54584780 IC50 = 1200 nM T59881 CH2GZ0 54584781 IC50 = 187 nM T59881 C0CRL3 54584782 IC50 = 2550 nM T59881 C98AJK 54584783 IC50 = 2 nM T59881 CHDO75 54584784 IC50 = 60 nM T59881 C14BIA 54584811 Ki > 10000 nM T59881 CHR91Z 54585227 Ki = 1.7 nM T59881 C8YD0H 54585429 Ki = 5.6 nM T59881 CQT40C 54585430 Ki = 20 nM T59881 C5N7VS 54585431 Ki = 1.2 nM T59881 CIJG06 54585709 IC50 > 20000 nM T59881 C3MQ4B 54585721 IC50 > 20000 nM T59881 CG6NT8 54585722 IC50 = 1044 nM T59881 CVR0A8 54585764 Ki = 560 nM T59881 CG7S2U 54585765 Ki = 790 nM T59881 CR5B8L 54585766 Ki = 430 nM T59881 C3MLH7 54586172 Ki >= 10000 nM T59881 CL79ME 54586390 Ki = 2.1 nM T59881 C1N7LU 54586391 Ki = 0.81 nM T59881 C60DIQ 54586392 Ki = 0.04 nM T59881 CAU1F5 54586482 IC50 = 60 nM T59881 CQT26P 54586699 IC50 = 52 nM T59881 C4Z9HU 54586715 IC50 = 500 nM T59881 CURC18 54586741 Ki > 10000 nM T59881 C73XTO 54586756 Ki = 2000 nM T59881 CXN6I1 54587400 Ki > 10000 nM T59881 C54PYE 54587727 IC50 > 20000 nM T59881 C9BSJ0 54587738 IC50 = 314 nM T59881 C56LJH 54587739 IC50 = 540 nM T59881 CP5KO4 54587779 Ki = 1000 nM T59881 CN13YR 54587780 Ki = 3200 nM T59881 CJ76VF 56657866 Ki = 282 nM T59881 C3T2HR 56657867 Ki = 66 nM T59881 CQG9J6 56657868 Ki = 87 nM T59881 C31CRV 56658409 EC50 = 15.85 nM T59881 C6T3VC 56658416 EC50 = 56 nM T59881 CJ5FQ4 56664848 Ki = 124 nM T59881 C5V3ME 56664849 Ki = 393 nM T59881 C3SYC9 56665377 EC50 = 15 nM T59881 CQN0G9 56668257 Ki > 10000 nM T59881 CL07IK 56671720 Ki = 126 nM T59881 CU9DK4 56671721 Ki > 1000 nM T59881 CSL0C7 56671723 Ki = 53 nM T59881 C8GLI4 56675151 Ki = 150 nM T59881 C05JPT 56678446 Ki > 10000 nM T59881 CNZU65 56682530 Ki = 0.42 nM T59881 CAG71L 57391220 Ki = 1154 nM T59881 C26OTQ 57394727 Ki = 1300 nM T59881 CFM91W 57399933 Ki > 1000 nM T59881 CHG37B 57519947 Ki = 9600 nM T59881 C0DB5C 57519948 Ki > 1000 nM T59881 C15NPY 57520031 Ki > 1000 nM T59881 C28VWF 68430068 Ki = 2 nM T59881 C7UGZ8 68430080 Ki = 9 nM T59881 C53WKC 68430310 Ki = 2 nM T59881 CLI79R 68430815 Ki = 84 nM T59881 CM61WS 68903270 Ki = 21 nM T59881 C2STV5 68905047 Ki = 36 nM T59881 C8M0XZ 68905061 Ki = 18 nM T59881 CL9R4M 68905198 Ki = 10 nM T59881 C3EKN9 68906357 Ki = 13 nM T59881 CS5C8Y 68907119 Ki = 32 nM T59881 C8S4AO 68907121 Ki = 58.5 nM T59881 CD1IQ4 70685417 Ki > 1000 nM T59881 CCTZ13 70685423 Ki > 1000 nM T59881 CUD97X 71451749 Ki > 10000 nM T59881 C7BCA6 71451750 Ki > 10000 nM T59881 CJGO63 71451752 Ki > 10000 nM T59881 C8KO3M 71453576 Ki > 10000 nM T59881 CG03VC 71455302 Ki > 10000 nM T59881 C0IZ5N 71457081 Ki > 10000 nM T59881 C1Q6RX 71462479 Ki > 10000 nM T59881 C2Y4UX 73348432 Ki = 1 nM T59881 C7GDP3 73350017 Ki = 0.78 nM T59881 C8GQK9 73350823 Ki > 10000 nM T59881 CQ8UO2 73351518 Ki = 1.2 nM T59881 CY4IW8 73351519 Ki = 0.43 nM T59881 CG8AD1 73354500 Ki = 4.8 nM T59881 CLMY01 76073634 EC50 > 10 nM T59881 CG0U7A 87451692 Ki = 1.1 nM T59881 C0Y1VJ 87451777 Ki = 0.9 nM T59881 C2WJ0B 87452314 Ki = 45 nM T59881 C1YLV9 90468623 EC50 = 170 nM T59881 CGZ9F1 90469608 EC50 = 64 nM T59881 CLXN70 90469674 EC50 = 110 nM T59881 CRO49T 90469675 EC50 = 140 nM T59881 CSKZ30 90469676 EC50 = 810 nM T59881 C3FE9W 118476329 EC50 = 210 nM T59881 CGKN68 118476331 EC50 = 480 nM T59881 C2TGY7 118476332 EC50 = 220 nM T59881 C4HGR0 118476333 EC50 = 580 nM T59881 CL2UK1 118476335 EC50 > 10000 nM T59881 C2G3FX 118476336 EC50 = 120 nM T59881 CR3O9G 118476337 EC50 = 160 nM T59881 C76ONJ 118476338 EC50 = 520 nM T59881 CC2UJ0 118476339 EC50 > 10000 nM T59881 CTV5Z6 118476341 EC50 = 350 nM T59881 C81BRW 118476342 EC50 > 10000 nM T59881 CRG4T1 118476343 EC50 = 140 nM T59881 C3YZ5M 118476344 EC50 > 10000 nM T59881 C24TBU 118476346 EC50 = 150 nM T59881 CEP13D 118476347 EC50 = 110 nM T59881 C2RE7I 118476348 EC50 = 330 nM T59881 C5E0HL 118476355 EC50 = 530 nM T59881 CUMW51 118476356 EC50 = 320 nM T59881 C21GNB 118476357 EC50 = 260 nM T59881 C6KZH9 118476358 EC50 = 480 nM T59881 C69TMC 118476359 EC50 = 150 nM T59881 C5Z9SC 118476360 EC50 = 380 nM T59881 C36WLI 118476361 EC50 = 40 nM T59881 CX9YV2 118476362 EC50 = 120 nM T59881 C94FHB 118476365 EC50 = 150 nM T59881 CI1E7V 118476366 EC50 = 190 nM T59881 CY4WD9 118476367 EC50 = 250 nM T59881 CS7DP0 118476369 EC50 > 10000 nM T59881 C7DAO4 118476383 EC50 = 140 nM T59881 C1KUY3 118476384 EC50 = 180 nM T59881 C5IFR0 118476385 EC50 = 46 nM T59881 C50MTE 118705579 Ki = 1.2 nM T59881 C9HX7Z 118705580 Ki = 149 nM T59881 CR3TZ0 118719818 EC50 = 700 nM T59881 CFG2V7 118719819 EC50 = 660 nM T59881 C4J6ZO 118719820 EC50 = 1000 nM T59881 C9B2WS 118719821 EC50 = 500 nM T59881 CAFX95 118719822 EC50 > 10 nM T59881 CH74ZW 118719823 EC50 > 10000 nM T59881 C7QI5K 118719824 EC50 = 1100 nM T59881 CAP85S 118719825 EC50 > 10000 nM T59881 CDR70N 118719826 EC50 > 10 nM T59881 CH0WU8 118719827 EC50 = 370 nM T59881 C1OMZ4 118719828 EC50 = 980 nM T59881 C72LOG 118719829 EC50 = 470 nM T59881 CD0P3Q 118719830 EC50 > 10000 nM T59881 CAKC58 118719831 EC50 = 2800 nM T59881 CIK48G 118719832 EC50 > 10000 nM T59881 CDSK02 118719833 EC50 = 260 nM T59881 C9GSF2 118719834 EC50 = 290 nM T59881 CS89AW 118719835 EC50 = 110 nM T59881 CTWG46 118719836 EC50 = 200 nM T59881 COQ71F 118719837 EC50 = 140 nM T59881 CT3LR1 118719838 EC50 = 440 nM T59881 CX3R0J 118719839 EC50 = 1800 nM T59881 CT3O7P 118719840 EC50 = 1300 nM T59881 CW2F8P 118719841 EC50 = 2600 nM T59881 CC9ZH4 118719842 EC50 = 590 nM T59881 C0LIH8 118719843 EC50 = 770 nM T59881 CYWM79 118719844 EC50 = 720 nM T59881 CGJ05D 118719845 EC50 = 240 nM T59881 CH3DE8 118720259 EC50 = 930 nM T59881 C3DLZ2 118720260 EC50 = 600 nM T59881 COD37S 118720261 EC50 > 10000 nM T59881 CPNB13 118720262 EC50 > 10000 nM T59881 CW4Q3B 118720263 EC50 > 10000 nM T59881 CI1SA4 118720264 EC50 = 3200 nM T59881 CX2K6O 118720265 EC50 = 830 nM T59881 COHG04 118720266 EC50 > 10000 nM T59881 CL2WY9 118720267 EC50 > 10000 nM T59881 C53KXO 118720268 EC50 = 7.7 nM T59881 CH2T3S 118720269 EC50 > 10000 nM T59881 C7KCE4 118720270 EC50 > 10000 nM T59881 CEK5A6 118720271 EC50 = 820 nM T59881 C4OSR7 118720272 EC50 = 450 nM T59881 C2Z8IG 118720273 EC50 > 10000 nM T59881 C3SD1R 118720274 EC50 > 10000 nM T59881 CXGF75 118720275 EC50 = 500 nM T59881 CZ96MR 118720276 EC50 = 3600 nM T59881 CM1V0E 118720277 EC50 = 1000 nM T59881 CJB1T7 118720278 EC50 = 100 nM T59881 C4KHJ3 118720279 EC50 = 100 nM T59881 C85IJS 118720280 EC50 = 440 nM T59881 CMK0A4 118720281 EC50 = 84 nM T59881 C1KPF5 118720282 EC50 = 87 nM T59881 C9XE0M 118720283 EC50 = 620 nM T59881 CXV09J 118720284 EC50 = 91 nM T59881 C2VF6Q 118720285 EC50 = 750 nM T59881 CLE5W1 118720286 EC50 = 160 nM T59881 C8QYZ7 118720287 EC50 = 1500 nM T59881 CMC18U 118720288 EC50 = 420 nM T59881 CF1RM4 118720289 EC50 = 190 nM T59881 CTS3Q9 118720290 EC50 = 850 nM T59881 C2T4QR 118734423 Ki = 12000 nM T59881 C7CNM8 132095331 EC50 = 130 nM T59881 CC09BD 135192928 IC50 = 59416 nM T59881 CWQ30S 135192932 IC50 = 27951 nM T59881 CSQ0Y2 135192979 IC50 = 56675 nM T59881 CQI48P 135192983 IC50 = 37562 nM T59881 CS8A2H 135192997 IC50 = 24540 nM T59881 CG3JX8 135193003 IC50 = 44436 nM T59881 CM26GP 135506374 Ki > 1000 nM T59881 C15WSK 136188833 IC50 = 387 nM T59881 C63UNT 145960494 EC50 = 2223 nM T59881 CIG1P6 145961670 Ki > 6000 nM T59881 C53JQB 145962220 EC50 = 2966 nM T59881 CRXH51 145963213 Ki > 6000 nM T59881 CQ2IG7 145976595 IC50 > 1000 nM T59881 CK04QR 145980069 Ki = 82 nM T59881 CH3B2Y 145980454 Ki = 45 nM T59881 CNRS86 145981524 Ki = 15.2 nM T59881 CW49CG 145983696 Ki = 8 nM T59881 C62UKO 145984883 Ki = 233 nM T59881 CSY72D 145987757 Ki = 104 nM T59881 CTN37Q 145988954 Ki = 30.2 nM T59881 CZV2L5 145991140 Ki = 41 nM T59881 C0B6JU 145991740 Ki = 47 nM T59881 C8PH6K 145993226 Ki = 192 nM T59881 CO4MS8 145993830 Ki = 1340 nM T59881 CC65HB 155513872 EC50 = 100 nM T59881 CSB84H 155515636 EC50 > 100000 nM T59881 CI4T0F 155518894 EC50 > 100000 nM T59881 C8BKV3 155523986 EC50 = 58 nM T59881 CDN37P 155524296 EC50 > 100000 nM T59881 C2RPD0 155527198 EC50 = 0.8 nM T59881 CA75ZF 155527876 EC50 > 100000 nM T59881 CYOF34 155532160 EC50 > 10 nM T59881 C8OT1G 155533728 EC50 > 100000 nM T59881 C2IZ6F 155535667 EC50 = 96 nM T59881 C4ZC5Y 155536940 EC50 = 0.5 nM T59881 CA6DC4 155542670 EC50 > 10000 nM T59881 C2JH0F 155555127 EC50 > 100000 nM T59881 COX4M3 155565903 EC50 > 10 nM T59881 D00SGZ 9917025 Ki = 25500 nM T59881 D01WHI 135413562 Ki = 3539 nM T59881 D09RIE 44419028 Ki = 1.2 nM T59881 D0K5NV 44428109 Ki > 1000 nM T59881 D0L0RP 44428107 Ki = 100 nM T59881 D0NC8V 6918854 Ki < 6309.57 nM T59881 D0R7QC 44419039 Ki = 0.37 nM T59881 D0W3IQ 44419025 Ki = 0.29 nM T59881 D0Y0SO 44419026 EC50 = 24 nM T59881 D0ZD0W 11366713 Ki = 0.49 nM T22285 D0I0DL 3689 IC50 = 39500 nM T22285 D02KLW 180081 IC50 = 29 nM T22285 D0K0DB 6604887 IC50 = 52000 nM T22285 C63KYD 66637 IC50 = 9700 nM T22285 CD48TY 694463 IC50 = 18600 nM T22285 C5Z6NT 3113150 IC50 = 19000 nM T22285 CXF09D 4231127 EC50 > 10000 nM T22285 CUGX54 9797385 EC50 > 10000 nM T22285 C8V2ZD 9799094 IC50 > 10000 nM T22285 CJ7Q4Y 9863769 IC50 > 10000 nM T22285 CAPM04 9927159 IC50 > 10000 nM T22285 CC9IL5 9928952 IC50 > 10000 nM T22285 C10ROQ 9972103 IC50 > 100000 nM T22285 C09KVR 9972180 IC50 > 100000 nM T22285 CGUQ10 10425979 IC50 > 100000 nM T22285 C4MCK2 10426105 IC50 > 100000 nM T22285 C3CID8 12045491 IC50 = 85000 nM T22285 C4Z0SE 12045492 IC50 = 77000 nM T22285 CN6RL1 12045493 IC50 = 77000 nM T22285 CJ0EZ4 12045494 IC50 > 100000 nM T22285 CM1S6P 12045495 IC50 = 73000 nM T22285 C13FGE 12045496 IC50 > 100000 nM T22285 CYL2J7 12045497 IC50 = 61000 nM T22285 CRB59C 12045498 IC50 = 64000 nM T22285 C27OQJ 12045832 IC50 > 100000 nM T22285 CH0RU2 20706422 IC50 > 10000 nM T22285 CI28HT 22432385 EC50 = 3200 nM T22285 CY0BC7 34924882 IC50 > 100000 nM T22285 CA72VD 44322229 IC50 = 62000 nM T22285 CQ21VN 44365962 IC50 = 35000 nM T22285 CDZ04W 44366039 IC50 = 75000 nM T22285 CCJD07 44366045 IC50 > 100000 nM T22285 C4BJ6F 44366056 IC50 > 100000 nM T22285 CR84AS 44366090 IC50 > 100000 nM T22285 C4DL5Q 44366109 IC50 > 100000 nM T22285 CRA24L 44366153 IC50 = 51000 nM T22285 C9CX5W 44366275 IC50 > 100000 nM T22285 CIC1G6 46861929 IC50 = 182000 nM T22285 C39CGI 56653056 EC50 = 100000 nM T22285 C4KWB0 56654447 EC50 = 28000 nM T22285 C7XPS1 66727815 IC50 = 1800 nM T22285 C6NX1P 118009615 EC50 = 8500 nM T22285 CL7P0F 118017713 EC50 = 2430 nM T22285 C1WV2M 155521371 IC50 = 198 nM T22285 CG3KS8 155557332 IC50 = 27 nM T22285 D06XGK 105074 EC50 = 21000 nM T22285 D07SGS 44292136 IC50 > 20000 nM T22285 D09HXX 4787937 IC50 = 110 nM T65889 C8VNO2 295161 EC50 > 20000 nM T65889 C6KH0U 711142 EC50 = 17300 nM T65889 CRXN16 746924 EC50 = 6900 nM T65889 CL7JG0 776870 IC50 = 100000 nM T65889 C64UHT 965237 EC50 = 18400 nM T65889 C6GQL8 2955824 EC50 > 20000 nM T65889 C7WN8Z 2988275 EC50 = 1500 nM T65889 CXBQ57 3638189 EC50 = 1100 nM T65889 C1WYZ0 3638190 EC50 = 16300 nM T65889 CG2C5N 3647906 EC50 = 410 nM T65889 CV6B5M 3647907 EC50 = 2000 nM T65889 CYE4D7 3648364 EC50 = 2200 nM T65889 CIV3P7 3656145 EC50 = 540 nM T65889 CK0J1O 3656150 EC50 = 1400 nM T65889 CN3CS7 4149969 EC50 = 11100 nM T65889 CG5UE2 4547230 EC50 = 790 nM T65889 C3UTE7 7066682 EC50 = 250 nM T65889 CRKT54 7066683 EC50 = 100 nM T65889 C8R0FJ 7601955 EC50 = 5200 nM T65889 CRQ20H 7601970 EC50 = 290 nM T65889 C09ZLQ 7720286 EC50 > 20000 nM T65889 C5SYH6 8015527 EC50 = 8300 nM T65889 C6PLG4 8087427 EC50 = 790 nM T65889 C4YKS1 8190555 EC50 = 18300 nM T65889 CPEM30 8512230 EC50 = 6000 nM T65889 CR7T5J 8512370 EC50 = 1300 nM T65889 CME23T 8512587 EC50 = 1300 nM T65889 CKR2P5 8512652 EC50 = 6400 nM T65889 C0RW7B 8516144 EC50 = 4600 nM T65889 C8Z6LB 8822317 EC50 = 940 nM T65889 CF4J7E 16615769 EC50 = 13400 nM T65889 CMY46P 20858997 EC50 = 4300 nM T65889 CCGY13 20969707 EC50 = 22 nM T65889 CLFY86 22518926 EC50 = 6000 nM T65889 C6TN5H 22548371 EC50 = 480 nM T65889 CGX7U9 22548477 EC50 = 260 nM T65889 C75VES 25417063 EC50 = 2300 nM T65889 C74JYC 44246498 EC50 = 73 nM T65889 C6U5XG 44246499 EC50 = 92 nM T65889 C41RNZ 44246502 EC50 > 20000 nM T65889 CN6H2U 44246503 EC50 > 20000 nM T65889 C7OV2M 44246504 EC50 > 20000 nM T65889 CBN97E 44543605 EC50 = 38 nM T65889 CVL82T 44623890 EC50 = 70 nM T65889 C2N4XY 44623893 EC50 = 13100 nM T65889 C1ZH9S 44623899 EC50 = 9000 nM T65889 CX34DM 44623900 EC50 > 20000 nM T65889 C7XIP5 44623901 EC50 = 10000 nM T65889 C89WYN 44623905 EC50 = 19900 nM T65889 C19KLY 44623906 EC50 = 210 nM T65889 C5LQ4C 44623907 EC50 > 20000 nM T65889 CTUD30 44623914 EC50 = 7100 nM T65889 CK3XB9 44623920 EC50 = 18300 nM T65889 C1UDT9 44623922 EC50 = 220 nM T65889 C3AR8W 44634848 EC50 = 210 nM T65889 CM3U6E 44634853 EC50 = 90 nM T65889 C86KJD 44634855 EC50 = 440 nM T65889 CN62ZM 44634859 EC50 = 140 nM T65889 C43MRY 44634865 EC50 = 560 nM T65889 CIS5W6 44634868 EC50 = 440 nM T65889 C43YJW 44634870 EC50 > 20000 nM T65889 CVA31W 46925978 EC50 = 570 nM T65889 CFW9K2 46925979 EC50 = 2100 nM T65889 C3WXG7 46925980 EC50 = 180 nM T65889 C7SF4R 46925981 EC50 = 3800 nM T65889 CGA51Q 46925984 EC50 = 510 nM T65889 CR9J8K 46925985 EC50 > 20000 nM T65889 CA6ZK3 46925986 EC50 = 230 nM T65889 C6TY5B 46925987 EC50 = 600 nM T65889 CNI4C5 46925988 EC50 = 240 nM T65889 COJ08B 46925989 EC50 = 90 nM T65889 C39FDP 46925991 EC50 = 880 nM T65889 C21OTY 46925992 EC50 = 170 nM T65889 CEC1B3 46926010 EC50 = 130 nM T65889 C5W7UY 46926011 EC50 = 290 nM T65889 C4MIF6 46926014 EC50 = 60 nM T65889 CQO7C8 57395381 EC50 = 6100 nM T65889 CUZ1K5 57398907 EC50 = 6600 nM T65889 CF51LO 57398908 EC50 = 7430 nM T65889 CR23IS 57398909 EC50 = 6100 nM T65889 CVZM95 71624854 EC50 = 70 nM T65889 CPO83E 91827688 IC50 = 95900 nM T65889 CSC4R1 131698387 IC50 = 16710 nM T65889 C7I0FG 145960470 IC50 = 2580 nM T65889 CK7PC4 145960501 IC50 > 20000 nM T65889 C3WGF0 145960585 IC50 = 9980 nM T65889 C0UXT7 145960872 IC50 > 20000 nM T65889 C3PKQ8 145960984 IC50 = 14110 nM T65889 CTW30D 145960988 IC50 = 15660 nM T65889 COL35X 145961254 IC50 = 1400 nM T65889 CC12OT 145961294 IC50 = 8780 nM T65889 C3O6BV 145961357 IC50 = 6790 nM T65889 CJFN52 145961746 IC50 = 5280 nM T65889 C83UNK 145961867 IC50 = 2210 nM T65889 CK3I6J 145961925 IC50 = 1740 nM T65889 CAP6O5 145962169 IC50 > 20000 nM T65889 CR4MK0 145962198 IC50 = 4230 nM T65889 C1K5BT 145962262 IC50 = 11700 nM T65889 CRUN17 145962267 IC50 > 20000 nM T65889 CT7NA8 145962307 IC50 = 8500 nM T65889 CM1EB8 145962338 IC50 = 5890 nM T65889 C20UKM 145962348 IC50 > 20000 nM T65889 CC9QJ7 145962375 IC50 > 20000 nM T65889 C3D1XG 145962426 IC50 = 4570 nM T65889 C0L3YC 145962579 IC50 > 20000 nM T65889 CG3VL1 145962648 IC50 = 4930 nM T65889 CS6TC3 145962785 IC50 = 14240 nM T65889 CPT25M 145962851 IC50 > 20000 nM T65889 CQZ6P2 145962864 IC50 > 20000 nM T65889 CH35RQ 145963014 IC50 > 20000 nM T65889 C0IX5E 145963290 IC50 > 20000 nM T65889 C3E7DG 145963371 IC50 = 5080 nM T65889 C90RBF 145963587 IC50 = 19730 nM T65889 C8RK1B 145963666 IC50 = 15240 nM T65889 C5BEN6 145968015 Ki = 50 nM T65889 C46KHV 145980165 IC50 = 880 nM T65889 CRJ30U 442279 EC50 = 6 nM T65889 D00LMG 5281697 IC50 = 12500 nM T03145 CAVF95 137553173 EC50 = 0.11 nM T03145 C7JT8X 145985109 IC50 = 45800 nM T03145 CVZ03D 145985495 IC50 = 49200 nM T67684 D01AZG 5073 Ki > 1000 nM T67684 D04JEE 4946 EC50 > 5011.87 nM T67684 D04LHJ 5459110 Ki = 0.1585 nM T67684 D08CTT 21855 Ki = 190.55 nM T67684 D09ZOQ 11519069 Ki = 0.06 nM T67684 D0B4TN 2381 Ki = 5.95 nM T67684 D0BZ7W 443879 Ki = 3.2 nM T67684 D0G8NN 119570 Ki > 10000 nM T67684 D0H3HM 60795 Ki > 1000 nM T67684 D0H7KF 5002 Ki > 1000 nM T67684 D0L4YD 154059 Ki = 13.18 nM T67684 D0M0AM 11693 IC50 = 0.2512 nM T67684 D0M6VK 71183 Ki = 0.1349 nM T67684 D0P1WA 5487427 Ki = 0.03162 nM T67684 D0Q9HF 187 EC50 = 3.2 nM T67684 D0RD5W 154417 Ki = 0.2692 nM T67684 D0RG3O 174174 Ki = 0.5 nM T67684 D0T0LM 4848 Ki = 47.86 nM T67684 D0U7BW 5831 EC50 = 70 nM T67684 D0V4QS 135398745 Ki = 100 nM T67684 D0VP1V 11434515 IC50 < 0.05012 nM T67684 D0Y5AM 444031 Ki = 0.84 nM T67684 D0Z1RV 135398737 Ki = 100 nM T67684 D04YEW 25147683 IC50 = 1.5 nM T67684 D05GNW 44517831 IC50 = 0.1585 nM T67684 D07EFM 2230 EC50 = 100 nM T67684 D0GP8P 10372836 IC50 = 1.585 nM T67684 D0I5XU 16065403 Ki = 0.128 nM T67684 D0K4HW 135409468 Ki = 90 nM T67684 D0LI1C 44469321 IC50 > 10000 nM T67684 D0N1HW 5311200 Ki > 10000 nM T67684 D0Z7AB 5487426 Ki = 0.2 nM T67684 D02JNY 10030021 Ki = 398.11 nM T67684 D06ACX 6436265 Ki = 93.33 nM T67684 D06DZI 107780 Ki < 1000 nM T67684 D08YVT 9894173 Ki = 700 nM T67684 D09FYQ 9577995 IC50 = 60 nM T67684 D0A2OW 107867 Ki = 2089 nM T67684 D0J8UV 9928284 EC50 = 5900 nM T67684 D0PZ9R 45260374 EC50 = 3.7 nM T67684 D0R1VL 132712 Ki = 776.25 nM T67684 D0VZ3D 129989 Ki = 63.1 nM T67684 C4AWJ9 2684 Ki = 2570.4 nM T67684 CKD46H 4022 Ki = 2398.83 nM T67684 C7VMZ3 4108 Ki = 277 nM T67684 C2AF8D 6060 EC50 = 220 nM T67684 CL53OW 6461 Ki = 2.6 nM T67684 C5H9CN 9287 Ki > 10000 nM T67684 CV42HF 16817 EC50 = 1000 nM T67684 C89UZB 18493 Ki = 4.25 nM T67684 CNZD18 36381 Ki = 336 nM T67684 CRCD50 60809 Ki = 7.762 nM T67684 C8E9XD 66007 IC50 = 26.3 nM T67684 C3WKC6 68835 IC50 = 87000 nM T67684 C3S8RF 71792 EC50 = 2696 nM T67684 C6ZQ4D 72064 Ki = 186 nM T67684 CA3W0P 100826 IC50 = 83000 nM T67684 CQA93V 118500 Ki = 780 nM T67684 CP9IQ0 160492 EC50 = 300 nM T67684 C2WO0V 163938 EC50 = 104000 nM T67684 CVWA68 197841 Ki = 270 nM T67684 CHLK79 214124 Ki = 9.9 nM T67684 C71KVJ 275176 Ki = 254 nM T67684 CD65GI 315401 Ki = 3.12 nM T67684 C1C2JH 372625 Ki = 10 nM T67684 C6OQ8S 410345 Ki = 8.37 nM T67684 CJ1QN5 425249 Ki = 59 nM T67684 C4J8NF 483747 Ki = 716 nM T67684 CX75UZ 598754 Ki > 19952.62 nM T67684 CQZ4A9 636934 Ki > 10000 nM T67684 CC56KR 639794 Ki = 15135.61 nM T67684 C91GCI 657308 Ki = 0.19 nM T67684 CEGR96 657346 Ki = 13489.63 nM T67684 CYO7F3 688566 IC50 = 0.9 nM T67684 C08WCU 851833 Ki > 19952.62 nM T67684 CO59NV 939077 IC50 = 0.76 nM T67684 CUD48J 952858 IC50 > 10000 nM T67684 CZ6Q4Y 1090198 IC50 > 10000 nM T67684 C4O6ZA 1090202 IC50 = 820 nM T67684 CWFV17 1392038 IC50 > 10000 nM T67684 CH5WR4 1421986 IC50 > 10000 nM T67684 C03LSA 1765112 IC50 = 1498 nM T67684 CPL49A 2157678 EC50 > 30000 nM T67684 CTRP25 2396803 Ki = 79.43 nM T67684 CS8N5X 2736067 Ki = 7943.28 nM T67684 CUF0Z9 3009352 Ki = 9089 nM T67684 CMK58I 3009353 Ki > 5300 nM T67684 CPN54Q 3009354 Ki > 5300 nM T67684 CG2PM5 3044806 IC50 = 1104000 nM T67684 C7ET2M 3156646 IC50 = 5600 nM T67684 C91XVY 3233138 IC50 > 1000 nM T67684 CJ6D8N 3342390 Ki < 1000 nM T67684 CI7DF6 3675988 Ki = 11481.54 nM T67684 C0YXV3 3676358 Ki > 10000 nM T67684 CX3S8T 4715419 Ki = 18197.01 nM T67684 C12BJA 4995951 Ki = 257.04 nM T67684 CS71UA 5189681 IC50 > 30000 nM T67684 CR5LG3 5310989 IC50 = 3704.2 nM T67684 C3A1FO 6604789 Ki = 50118.72 nM T67684 CFN7L4 6604866 Ki = 138.04 nM T67684 C2IP0Y 7022778 Ki = 43651.58 nM T67684 CVSC58 7047822 Ki = 25118.86 nM T67684 C32TSZ 7141654 Ki = 147910.84 nM T67684 C7NJZ2 7141656 Ki = 12022.64 nM T67684 CU3W4K 9044803 IC50 = 27542.29 nM T67684 CYH05F 9794266 Ki = 830 nM T67684 CEDB68 9798900 IC50 = 6 nM T67684 CL94XF 9799291 Ki = 3.7 nM T67684 C7MBO3 9809330 Ki = 5.012 nM T67684 CMC3O6 9821459 Ki = 4.2 nM T67684 C6NJO3 9827782 Ki = 3.7 nM T67684 CH74OS 9846311 Ki = 2.8 nM T67684 C3YI2L 9857572 IC50 = 4.3 nM T67684 C1N0KW 9867847 Ki = 0.48 nM T67684 CA43HC 9874175 Ki = 0.01 nM T67684 CZHS28 9880462 Ki = 0.63 nM T67684 CJ5K1D 9889312 Ki = 29.4 nM T67684 CR5PO3 9903030 IC50 = 74.7 nM T67684 CUN81Q 9905249 Ki > 10000 nM T67684 C2U5LK 9905467 IC50 = 155.8 nM T67684 CCT20X 9905731 Ki = 11 nM T67684 CYWQ50 9906447 Ki = 204 nM T67684 CDB9E1 9909907 Ki = 79.43 nM T67684 CL5HA4 9910802 Ki = 3.2 nM T67684 CXAV92 9911615 Ki = 229.09 nM T67684 CXAY37 9913341 Ki = 25.12 nM T67684 C24PKZ 9913892 Ki = 7.943 nM T67684 C3L5GV 9928017 IC50 = 0.6 nM T67684 CRV17M 9931930 Ki = 70.79 nM T67684 C50NSR 9936450 Ki = 2.884 nM T67684 CSH40U 9936494 IC50 = 2070 nM T67684 C65PMK 9944783 IC50 = 1.7 nM T67684 C36NIB 9946010 IC50 = 1 nM T67684 CKQM18 9946298 Ki = 0.25 nM T67684 CY4L1D 9946632 IC50 = 15 nM T67684 CFG21X 9966959 IC50 = 17.7 nM T67684 CH23EP 9967590 IC50 = 1.2 nM T67684 CYNT43 9968046 Ki = 2089.3 nM T67684 CQF52V 9969695 Ki = 10 nM T67684 CCM72P 9974222 IC50 = 100.7 nM T67684 C3G0VC 9985181 Ki = 46.4 nM T67684 CB8VU6 9986442 Ki = 0.32 nM T67684 C9XS0E 9990434 EC50 = 16400 nM T67684 CYK1U4 9996901 IC50 = 110 nM T67684 C9FR0C 9998508 Ki = 1698.24 nM T67684 CQL12P 10004545 Ki > 2000 nM T67684 CK19GL 10007637 IC50 = 0.7 nM T67684 CV7R9F 10020040 Ki > 10000 nM T67684 CU4Z8L 10020681 IC50 = 1069.4 nM T67684 CQZ0K4 10027177 EC50 > 50000 nM T67684 C7I6DA 10035281 Ki = 15000 nM T67684 CBJ63D 10043954 Ki = 1737.8 nM T67684 CPCL60 10044685 Ki = 25.12 nM T67684 CQ8F9I 10049361 Ki = 1 nM T67684 C56FEU 10053613 IC50 = 2 nM T67684 CR73MA 10054373 Ki = 0.14 nM T67684 C9OQ2S 10066369 Ki = 2238.72 nM T67684 CI6SD7 10066972 Ki = 2089.3 nM T67684 CCO72H 10082470 IC50 = 1600 nM T67684 C8NQ3I 10092649 Ki = 430 nM T67684 CU25MW 10109130 Ki = 0.05 nM T67684 CIN03S 10109563 Ki = 0.3162 nM T67684 CG0O9Z 10109893 Ki = 316.23 nM T67684 CUT05R 10114698 Ki = 457.09 nM T67684 C9XDU8 10119938 IC50 = 0.5 nM T67684 C9WXO8 10130070 EC50 = 8900 nM T67684 C20GMN 10132599 IC50 = 3.6 nM T67684 CFH60N 10133281 IC50 = 5.9 nM T67684 C90FZG 10139614 Ki = 281.84 nM T67684 C0PO3J 10142923 Ki = 25.12 nM T67684 CPF96U 10143717 IC50 = 0.3 nM T67684 CC8YJ1 10143857 IC50 = 0.6 nM T67684 C7LP4V 10143953 IC50 = 1.62 nM T67684 CYU79M 10143955 Ki = 0.07 nM T67684 C9DY4P 10155225 Ki = 2.512 nM T67684 CDOI12 10155850 Ki = 1.995 nM T67684 CG78WP 10160073 Ki = 151 nM T67684 CZ8E9X 10160219 Ki = 100 nM T67684 CVI4O6 10164136 IC50 = 0.8 nM T67684 CXCT70 10165876 IC50 = 0.2 nM T67684 CGA94F 10171570 Ki = 50 nM T67684 C5WO3U 10171655 Ki = 15.85 nM T67684 C4TR5Q 10180872 Ki = 0.97 nM T67684 C1B8RO 10187215 IC50 = 0.6 nM T67684 CI2A5S 10193005 Ki = 10 nM T67684 CS5TJ2 10193093 Ki = 6.3 nM T67684 CO05SP 10199963 Ki = 0.79 nM T67684 COR14Y 10203251 Ki = 70.79 nM T67684 CB69ND 10204457 Ki = 6.8 nM T67684 CUW93D 10208896 IC50 = 0.3 nM T67684 C57WMS 10208971 IC50 = 1 nM T67684 CB35LH 10214932 Ki = 20 nM T67684 CJ5V2S 10225340 Ki = 13.76 nM T67684 C04QCB 10225881 Ki = 338.84 nM T67684 C6A5KD 10226456 Ki = 125.89 nM T67684 C8XY5N 10229166 IC50 = 0.6 nM T67684 C0TD1V 10236397 Ki = 16 nM T67684 C6CN3D 10236419 Ki = 79 nM T67684 C4R8YW 10236511 Ki = 25 nM T67684 CO64WJ 10236758 Ki = 1202.26 nM T67684 CRQ8D4 10240891 EC50 = 14600 nM T67684 C49MUR 10246307 IC50 = 1.1 nM T67684 C3QGA5 10251795 EC50 > 50000 nM T67684 CW90FO 10261985 EC50 = 130 nM T67684 C1FCP7 10262466 Ki = 392 nM T67684 CH31DX 10267394 Ki > 10000 nM T67684 CC6RP7 10267601 IC50 = 40.8 nM T67684 CT07QH 10269503 Ki = 0.1995 nM T67684 CFN5O4 10269504 Ki = 3.2 nM T67684 CCN9B4 10269809 Ki = 15.85 nM T67684 CY3E5J 10274019 Ki = 0.16 nM T67684 C8HD7O 10291366 Ki = 0.1259 nM T67684 C6N9XM 10291977 Ki = 0.08 nM T67684 C7WMZ6 10300660 IC50 = 0.8 nM T67684 CU89JD 10314060 Ki > 10000 nM T67684 CD1C0H 10315426 Ki = 3311.31 nM T67684 CG14VC 10326800 Ki = 0.18 nM T67684 C0U7AV 10327461 Ki = 0.1995 nM T67684 C9NQ0K 10327462 Ki = 0.1995 nM T67684 C3E5CB 10337773 Ki = 31622.78 nM T67684 C0DTX5 10348864 Ki = 0.14 nM T67684 C6S7GK 10354348 IC50 > 100000 nM T67684 C7BZ1R 10358345 IC50 = 349 nM T67684 CBSA40 10360219 Ki = 1621.81 nM T67684 CXI91M 10372344 Ki = 0.07943 nM T67684 CY9G0R 10375322 EC50 = 9600 nM T67684 C72EML 10392704 IC50 = 33.4 nM T67684 CR0V3S 10394806 Ki = 0.3162 nM T67684 C85QEA 10397133 EC50 = 8400 nM T67684 C5TX2E 10397356 EC50 = 8800 nM T67684 CL7D2U 10421982 Ki = 3200 nM T67684 CA63EB 10438748 Ki = 0.74 nM T67684 CA4PR8 10439505 Ki = 0.631 nM T67684 C5BEJ0 10442081 EC50 = 620 nM T67684 CIRS06 10442337 EC50 = 500 nM T67684 CDV2K0 10460513 IC50 = 599.3 nM T67684 C6JY9O 10461973 Ki = 0.1 nM T67684 CC9AV4 10465280 EC50 = 140 nM T67684 C53SCK 10468535 Ki = 100 nM T67684 CEF2O6 10478367 Ki > 10000 nM T67684 CRP7L9 10484263 Ki = 7.5 nM T67684 CC3Z2P 10484922 Ki = 1.585 nM T67684 C1GT3O 10487582 IC50 = 380 nM T67684 C8COH6 10499832 IC50 = 2046.8 nM T67684 C18ZYN 10500741 Ki = 2.5 nM T67684 CU0B8N 10501523 Ki = 220 nM T67684 CO62HL 10503358 Ki = 2 nM T67684 CS1P4M 10511551 IC50 = 1200 nM T67684 CP9M5J 10516408 IC50 = 2312.2 nM T67684 C37PDA 10518821 IC50 = 16753.5 nM T67684 C6T1JW 10521205 IC50 = 529.6 nM T67684 C4WZ3R 10522202 IC50 = 2801.3 nM T67684 C5MB2F 10522336 IC50 = 1600.8 nM T67684 C3EZ5Y 10525412 Ki = 6.4 nM T67684 C0K9HN 10538337 IC50 = 88401.3 nM T67684 C3Y6JB 10546275 IC50 = 201.6 nM T67684 CI3GQ6 10547222 IC50 = 983 nM T67684 C6XKZ9 10549581 IC50 = 871.1 nM T67684 CSC81Z 10551354 Ki = 3.1 nM T67684 CFD40Z 10567192 IC50 = 299.3 nM T67684 C4AL8Q 10569816 IC50 = 1491 nM T67684 CHI03M 10572657 Ki = 100 nM T67684 C0Z5PY 10572658 Ki = 190 nM T67684 CV62YH 10573458 Ki = 11 nM T67684 CB37SH 10573693 IC50 = 5051.5 nM T67684 CR2GX4 10574041 Ki = 30 nM T67684 C71VMD 10591874 IC50 = 211.3 nM T67684 C94VUE 10592484 IC50 = 1095.5 nM T67684 C51LBK 10593954 IC50 = 1244.3 nM T67684 CH2QU8 10594386 IC50 = 24861.7 nM T67684 CY54RA 10595006 Ki = 1370 nM T67684 C6VGM0 10597259 Ki = 19 nM T67684 CVY63G 10598540 Ki = 93 nM T67684 CZRJ60 10610375 IC50 = 5523.7 nM T67684 CX01SE 10611310 IC50 = 1689.3 nM T67684 CO3H7D 10614695 IC50 = 4069.7 nM T67684 C3BK2J 10619926 Ki = 50 nM T67684 C34LMA 10621363 Ki = 2.3 nM T67684 CSGO98 10622033 Ki = 6.2 nM T67684 C92HRJ 10622718 Ki = 18 nM T67684 CLJ29W 10623721 Ki = 21 nM T67684 CJL4R1 10636001 IC50 = 684 nM T67684 C09XHV 10638050 IC50 = 918 nM T67684 C5VWL8 10641009 IC50 = 114.7 nM T67684 C2ZTE6 10646906 Ki = 7.8 nM T67684 CDAG26 10646948 Ki = 5.4 nM T67684 CZ7M1D 10647553 Ki = 17 nM T67684 CX49UY 10647703 Ki = 6.1 nM T67684 CONH15 10663572 IC50 = 403.6 nM T67684 C6WQ2Z 10664532 IC50 = 1653.8 nM T67684 C8CF4H 10666533 IC50 = 1218.7 nM T67684 C56EGM 10670917 Ki = 6.9 nM T67684 C1DSK6 10670961 Ki = 15 nM T67684 CUYW18 10671167 Ki = 28 nM T67684 C0AV8X 10678449 IC50 = 2200 nM T67684 C32KQX 10684720 IC50 = 535.5 nM T67684 C32EGP 10686988 IC50 = 220.3 nM T67684 C9O6LN 10688349 IC50 = 3175.4 nM T67684 C6PDH5 10693031 Ki = 3.5 nM T67684 C62MCG 10716120 Ki = 11 nM T67684 CS3W1G 10718110 Ki = 8.9 nM T67684 CEB3A5 10726038 IC50 = 300 nM T67684 C5OF4K 10739662 Ki = 17 nM T67684 CGFV60 10742178 Ki = 1000 nM T67684 CC21XD 10755732 IC50 = 290 nM T67684 CHL29Z 10755733 IC50 = 257.5 nM T67684 C4JXA3 10757736 IC50 = 2551.1 nM T67684 CPQ7Z3 10760249 IC50 = 88 nM T67684 C5P3DQ 10761219 IC50 = 14309.6 nM T67684 CX4LT3 10777692 IC50 = 6874.7 nM T67684 CA4QI2 10782321 IC50 = 6712.1 nM T67684 C4N9IT 10782462 IC50 = 109.6 nM T67684 C6FC0M 10784004 IC50 = 749.3 nM T67684 CV8TE0 10785471 IC50 = 399.5 nM T67684 CLI6Z3 10789183 Ki = 1.995 nM T67684 CW5TJ6 10797864 IC50 = 28 nM T67684 C9SEA6 10806268 IC50 = 162.5 nM T67684 CGR64V 10808719 IC50 = 1842 nM T67684 C3QK4R 10810094 Ki = 270 nM T67684 CR4XK8 10812455 Ki = 3.8 nM T67684 CK1D3J 10827157 IC50 = 844.6 nM T67684 CR1X5L 10829928 IC50 = 1927.8 nM T67684 C0GS8Z 10830843 Ki = 320 nM T67684 C2M0QO 10834711 Ki = 3.6 nM T67684 C27NPT 10835518 Ki = 12 nM T67684 C2S6DG 10836338 Ki = 13 nM T67684 CB7E2O 10846833 IC50 = 9700 nM T67684 CAG97P 10851461 Ki = 46 nM T67684 CH9WK6 10851853 IC50 = 356.9 nM T67684 CX6AP3 10852843 IC50 = 4514.2 nM T67684 C5PRT6 10854879 IC50 = 675.6 nM T67684 C8HI5L 10854880 IC50 = 86.5 nM T67684 CZ85AJ 10862395 Ki = 91.2 nM T67684 CHE9P4 10865439 Ki = 97.2 nM T67684 CCM3L9 10870954 Ki = 23988.33 nM T67684 C2YNC5 10871551 Ki = 281.84 nM T67684 CFAD04 10874119 Ki = 1380.38 nM T67684 CTV95B 10880435 Ki = 1548.82 nM T67684 C4A8QE 10916286 Ki = 5128.61 nM T67684 CQLR32 10919522 Ki = 0.25 nM T67684 CC12TE 10925451 Ki = 501.19 nM T67684 C5LVY0 10949838 Ki = 218.78 nM T67684 CE05FM 10951142 Ki = 50.12 nM T67684 C3K6JV 10957754 Ki = 575.44 nM T67684 CN4QT5 10963509 Ki = 422 nM T67684 C4WV8L 10969390 Ki = 707.95 nM T67684 CTYZ13 10969696 Ki = 2754.23 nM T67684 C41PXY 10982070 Ki = 398.11 nM T67684 C9E2MP 10984804 Ki = 99 nM T67684 C2W3GM 11000399 Ki = 11748.98 nM T67684 C6NH9T 11001809 Ki = 8128.31 nM T67684 CQ8D4K 11004046 Ki = 912.01 nM T67684 C6BG1N 11006792 Ki = 2.2 nM T67684 CU4Z0J 11011332 Ki = 8128.31 nM T67684 CZK86F 11011757 Ki = 288.4 nM T67684 CVA6U9 11012653 Ki = 1819.7 nM T67684 CPM1Z7 11012712 Ki = 1174.9 nM T67684 CW23BJ 11013666 Ki = 67.61 nM T67684 C6TF5I 11015312 Ki = 1023.29 nM T67684 C7Y1DO 11024241 Ki = 1047.13 nM T67684 C3L9ON 11034265 Ki = 263.03 nM T67684 CHDT49 11039424 Ki = 0.31 nM T67684 CP9OJ6 11045444 Ki = 630.96 nM T67684 C4ZUH9 11048067 Ki = 263.03 nM T67684 CQ8O3Y 11057942 Ki = 25703.96 nM T67684 CIG31V 11061341 Ki = 0.47 nM T67684 CT3XN5 11071537 Ki = 79.43 nM T67684 C5VQ6H 11079969 Ki = 407.38 nM T67684 CWS56C 11092603 Ki = 676.08 nM T67684 C02MPO 11099206 Ki = 1905.46 nM T67684 CSNA03 11101362 Ki = 2754.23 nM T67684 CF81CB 11110049 Ki = 134896.29 nM T67684 C7ROJ1 11112362 Ki = 2041.74 nM T67684 C9CY0M 11120347 Ki = 501.19 nM T67684 C2C4AN 11131099 Ki = 3162.28 nM T67684 C1T9WI 11143997 Ki = 229.09 nM T67684 C4JS0X 11168935 IC50 = 5.012 nM T67684 CWN95Y 11191775 IC50 < 10 nM T67684 C9WS8C 11215075 IC50 = 50.12 nM T67684 CX69QO 11223597 Ki = 0.45 nM T67684 C32PXU 11235699 IC50 < 10 nM T67684 C9X7AO 11249473 IC50 = 50.12 nM T67684 C0ZM4H 11271303 IC50 < 10 nM T67684 CA6O9B 11272761 IC50 < 10 nM T67684 CXBP81 11273131 IC50 = 31.62 nM T67684 CR7L6F 11284402 IC50 = 6.31 nM T67684 CI1EN4 11306851 IC50 = 1.68 nM T67684 CBR60Z 11318734 IC50 = 31.62 nM T67684 C96RYX 11330061 IC50 = 100 nM T67684 CN3YR6 11341753 IC50 = 10 nM T67684 C80ANS 11341940 IC50 = 10 nM T67684 C64UOJ 11364721 IC50 = 10 nM T67684 C6FA7M 11398061 IC50 = 89.6 nM T67684 C3B1WK 11398832 IC50 = 501.19 nM T67684 CQB9T8 11399125 IC50 = 3981.07 nM T67684 CJ6U1L 11410317 IC50 = 79.43 nM T67684 C01CUI 11410490 IC50 = 50.12 nM T67684 CA1VK2 11421571 IC50 = 316.23 nM T67684 C85LYP 11430418 IC50 > 1000 nM T67684 C9FNM4 11431811 Ki = 0.0098 nM T67684 CGD57K 11431873 Ki = 0.16 nM T67684 CLP2R9 11431874 IC50 < 10 nM T67684 C9NUV4 11442477 IC50 = 1 nM T67684 C2ME0L 11442668 IC50 < 10 nM T67684 CBO07Q 11442669 IC50 = 26.3 nM T67684 C50QGB 11443944 IC50 = 79.43 nM T67684 CQT8K2 11455956 IC50 = 19.95 nM T67684 CIN42A 11489418 IC50 = 0.39 nM T67684 CTVZ02 11503335 IC50 = 3 nM T67684 CFSH67 11504490 Ki = 0.03162 nM T67684 CBZ5E8 11508710 IC50 = 22.9 nM T67684 CSP02B 11510357 IC50 = 16 nM T67684 CF4H0Y 11512118 IC50 < 10000 nM T67684 CGCF61 11515738 Ki < 100000 nM T67684 CXE30W 11517306 IC50 = 486000 nM T67684 C7OKD1 11518067 IC50 = 2.3 nM T67684 C5CXG8 11519317 IC50 < 10000 nM T67684 CY63VP 11523050 Ki = 33884.42 nM T67684 C07AJD 11530306 Ki < 100000 nM T67684 CRX7T9 11531768 IC50 = 208000 nM T67684 C89JTB 11532924 Ki = 160 nM T67684 CJP9L7 11533794 IC50 < 10000 nM T67684 CE6HA5 11539228 IC50 = 135000 nM T67684 CWUP85 11542982 Ki < 100000 nM T67684 CZBJ25 11545844 IC50 = 104000 nM T67684 C6B2XK 11547052 IC50 = 11.3 nM T67684 CNZJ38 11552174 IC50 = 10.9 nM T67684 C01HAQ 11557048 IC50 = 3.981 nM T67684 CP9UJ1 11569907 IC50 = 0.31 nM T67684 CP04FM 11569925 IC50 = 17.7 nM T67684 C4DL2I 11578568 IC50 = 1995.26 nM T67684 CYW90N 11583261 IC50 = 2.8 nM T67684 C6D1MA 11584660 IC50 = 3162.28 nM T67684 C4TN9E 11585116 IC50 < 10000 nM T67684 CEHP14 11586481 Ki < 100000 nM T67684 CP3Y7J 11588240 Ki < 100000 nM T67684 CM0KX9 11592004 IC50 < 10000 nM T67684 CP3G5L 11602980 IC50 = 7.2 nM T67684 CQAU82 11606546 IC50 = 39000 nM T67684 C15DMA 11617374 IC50 = 27.5 nM T67684 CE07UT 11619197 IC50 = 4.6 nM T67684 CQ5PI4 11622544 Ki < 100000 nM T67684 CK4GS9 11626846 IC50 = 6.4 nM T67684 C6E5GV 11633225 IC50 < 10 nM T67684 CE0K7I 11633398 IC50 = 30000 nM T67684 C03UGR 11635209 IC50 < 10000 nM T67684 CHQ19E 11642406 IC50 < 10000 nM T67684 COFE39 11649605 IC50 < 10000 nM T67684 CF2ZC0 11651360 Ki < 100000 nM T67684 CHKN81 11653111 Ki < 100000 nM T67684 C27XOS 11660220 Ki < 100000 nM T67684 C27WBZ 11664152 IC50 = 17000 nM T67684 C0N4BQ 11672895 Ki < 100000 nM T67684 C8Q5WO 11674313 Ki = 49 nM T67684 C0ZK8U 11678377 IC50 = 0.8 nM T67684 CN4Z5C 11679149 IC50 > 10000 nM T67684 CI5B1R 11690967 IC50 = 2 nM T67684 CTWG21 11691470 IC50 = 87000 nM T67684 CQD96L 11691949 Ki = 0.13 nM T67684 C25DBM 11692149 IC50 = 9500 nM T67684 CW8CE2 11694118 Ki < 100000 nM T67684 CF8MO2 11694119 Ki < 100000 nM T67684 CMT6F0 11695697 IC50 = 37.3 nM T67684 CZIX30 11699451 IC50 = 12000 nM T67684 C5XN4V 11705919 IC50 < 10000 nM T67684 CY31MF 11712407 IC50 = 21.2 nM T67684 C5XU0N 11714747 IC50 = 199.53 nM T67684 C9BF1S 11715398 Ki < 100000 nM T67684 CWE71N 11718536 Ki = 1.9 nM T67684 C0O2QC 11725334 IC50 = 2.2 nM T67684 CEY7J3 11729182 Ki = 15488.17 nM T67684 CPG15O 11743399 IC50 > 1000 nM T67684 C4QVR6 11748799 Ki = 25.7 nM T67684 CQLP36 11759058 Ki = 48977.88 nM T67684 CW3GA7 11759212 Ki = 95.5 nM T67684 CBM05D 11759379 Ki = 1778.28 nM T67684 CFZ4L5 11767229 Ki = 1 nM T67684 C39HRB 11793999 IC50 = 447.9 nM T67684 CM16WE 11794901 Ki = 14 nM T67684 CT8P7Q 11796409 Ki = 16 nM T67684 C91DQM 11796509 Ki = 5.9 nM T67684 CHEA80 11798126 Ki = 3.5 nM T67684 CT4F2C 11808040 Ki = 31.62 nM T67684 CXQ10I 11808946 Ki = 309.03 nM T67684 C6EXD3 11808947 Ki = 741.31 nM T67684 C30WRH 11809446 Ki = 8912.51 nM T67684 CJIA51 11828362 Ki = 0.76 nM T67684 CR9FJ2 11833737 Ki = 2511.89 nM T67684 CZ3AX9 11834199 Ki = 954.99 nM T67684 C85LXI 11857427 Ki = 0.05012 nM T67684 C8JQL7 11957735 IC50 > 10000 nM T67684 CL91TM 11968014 Ki = 6.5 nM T67684 C5P3XD 12586122 Ki > 50000 nM T67684 CR10FQ 13567080 Ki = 1.778 nM T67684 CWP60M 13621534 EC50 > 50000 nM T67684 CL8G7N 13621544 EC50 = 1800 nM T67684 CBS93C 13621546 EC50 = 3400 nM T67684 C7NL5D 13621548 EC50 > 50000 nM T67684 C8GDT6 13621550 EC50 > 50000 nM T67684 CEGU40 13621552 EC50 > 50000 nM T67684 C38UXQ 13621554 EC50 > 50000 nM T67684 CE12ZW 13621556 EC50 = 13000 nM T67684 CR91KI 13621558 EC50 > 50000 nM T67684 CTCX78 13621560 EC50 > 50000 nM T67684 C63DUH 13621562 EC50 = 1200 nM T67684 C5PRZ0 13621564 EC50 > 50000 nM T67684 CV21AW 13621566 EC50 = 4500 nM T67684 C18PKQ 13621568 EC50 = 800 nM T67684 C7UE4K 13621570 EC50 = 1600 nM T67684 C1GE5A 13621573 EC50 = 20000 nM T67684 C0O8JQ 13621575 EC50 > 50000 nM T67684 COT9Z6 13981863 Ki = 2.11 nM T67684 C1IDP8 13981864 Ki = 28 nM T67684 C19BYU 14479864 IC50 < 1 nM T67684 CS54WY 14537188 Ki = 52.2 nM T67684 CA87RQ 14660293 IC50 = 100000 nM T67684 CMO81H 14925759 Ki = 17782.79 nM T67684 CZ16XJ 15157137 Ki = 1.7 nM T67684 C5VC9Z 15157138 Ki = 4 nM T67684 C7VT5X 15157139 Ki = 31.2 nM T67684 CD3MI7 15157140 Ki = 160 nM T67684 CY80DC 15157141 Ki = 178 nM T67684 C9C6WP 15629515 Ki = 28000 nM T67684 CIW40C 15888010 Ki = 5.1 nM T67684 CJKM40 15888011 Ki = 1.4 nM T67684 CT64BE 15945874 IC50 = 19.95 nM T67684 C9NS7T 15951516 IC50 < 10000 nM T67684 CZ8BL1 16034837 Ki = 0.18 nM T67684 CUB5X2 16038385 EC50 > 10000 nM T67684 CM7FS0 16041938 IC50 < 10000 nM T67684 CL1CM4 16065135 Ki = 0.25 nM T67684 CI1QH2 16065136 Ki = 1.6 nM T67684 C9CU8F 16065137 Ki = 0.201 nM T67684 CCS3K1 16065268 Ki = 0.27 nM T67684 CEZ9Y0 16065269 Ki = 2.3 nM T67684 CVZ68N 16065402 Ki = 0.049 nM T67684 CJE56L 16065404 Ki = 1.9 nM T67684 C45DKH 16065405 Ki = 0.6 nM T67684 CW58VJ 16065406 Ki = 0.73 nM T67684 CCEH96 16065407 Ki = 0.163 nM T67684 C2D8RK 16065541 Ki = 0.71 nM T67684 CO25RH 16065543 Ki = 0.22 nM T67684 CZ47FJ 16071018 EC50 = 2511.89 nM T67684 C3T0UX 16085999 Ki = 0.48 nM T67684 CWI32N 16086000 Ki = 0.51 nM T67684 C71HBL 16086001 Ki = 0.17 nM T67684 C7EM1G 16086003 Ki = 4.2 nM T67684 CFU72Z 16086004 Ki = 3.7 nM T67684 CTOM27 16086005 Ki = 1.2 nM T67684 C7LBY9 16086015 Ki = 150 nM T67684 CTH0Y3 16086017 Ki = 49 nM T67684 CP5H4W 16086021 Ki = 23 nM T67684 C50THR 16086031 Ki = 29 nM T67684 CBK05F 16086035 Ki = 170 nM T67684 CLW4I8 16086039 Ki = 48 nM T67684 C7WF9Y 16086059 Ki = 0.3 nM T67684 C05YVJ 16086060 Ki = 0.39 nM T67684 CMQ8U3 16086061 Ki = 0.92 nM T67684 CEI8G1 16086062 Ki = 0.53 nM T67684 CGB89M 16086063 Ki = 0.19 nM T67684 CUS73E 16086064 Ki = 0.51 nM T67684 CHJ07L 16086065 Ki = 2.8 nM T67684 CEV68D 16086066 Ki = 0.39 nM T67684 CIX9M7 16086067 Ki = 1.6 nM T67684 C1XZ7V 16094783 Ki = 50.12 nM T67684 CO16DS 16094788 Ki = 1584.89 nM T67684 CYN71L 16094791 Ki = 251.19 nM T67684 C2HK7W 16094793 Ki = 199.53 nM T67684 C9R0JN 16094810 Ki = 199.53 nM T67684 CTYI57 16115796 Ki = 2.455 nM T67684 C5HSD9 16115797 Ki = 2.188 nM T67684 CQ85FK 16115798 Ki = 1.698 nM T67684 CR1Z4N 16115799 Ki = 1.445 nM T67684 CLA6E0 16115800 Ki = 5.012 nM T67684 CTE0R7 16115942 Ki = 4.898 nM T67684 C7IC9E 16115944 Ki = 0.5888 nM T67684 CQ3C9X 16115946 Ki = 0.912 nM T67684 C0JGY1 16115950 Ki = 5.248 nM T67684 CZ67DO 16115951 Ki = 0.8913 nM T67684 CO3YU4 16116082 Ki = 0.7413 nM T67684 C3IKJ0 16116084 Ki = 0.3388 nM T67684 CWU6P3 16123945 EC50 = 3981.07 nM T67684 C6B4YR 16124705 Ki = 6.59 nM T67684 C42YXI 16124706 Ki = 1.72 nM T67684 CY0KP2 16124707 Ki = 2.75 nM T67684 C7RN3Z 16124708 Ki = 18.5 nM T67684 C8RVY4 16124710 Ki = 16.8 nM T67684 CZ7JF4 16124769 Ki = 26.8 nM T67684 CJ5GP8 16125158 Ki = 2185 nM T67684 CI1G8P 16125223 Ki = 13.3 nM T67684 CO24GD 16125224 Ki = 114 nM T67684 CRW9N0 16125257 Ki = 249 nM T67684 CK1OD5 16125325 Ki = 310 nM T67684 CG76PT 16125327 Ki = 3158 nM T67684 CT04HJ 16125329 Ki = 2065 nM T67684 CXY50Q 16125331 Ki = 0.7 nM T67684 CA05KV 16125335 Ki = 6.66 nM T67684 C1DZA2 16125369 Ki = 2445 nM T67684 C5G6IH 16125370 Ki = 0.96 nM T67684 CGUF57 16125371 Ki = 82 nM T67684 C0J6CH 16125372 Ki = 2.8 nM T67684 C9YJT7 16125373 Ki = 2.57 nM T67684 C75NYZ 16125374 Ki = 2.7 nM T67684 CN5LU9 16125398 Ki = 7.6 nM T67684 CNHJ78 16125400 Ki = 3.01 nM T67684 CP31TE 16125437 Ki = 152 nM T67684 CD9NV1 16125443 Ki = 923 nM T67684 C7L1QR 16125444 Ki = 101 nM T67684 C8O3YT 16125470 Ki = 612 nM T67684 C8J3YQ 16125503 Ki = 354 nM T67684 CE8G4T 16125505 Ki = 117 nM T67684 CVA18O 16125506 Ki = 1630 nM T67684 CQV41Z 16125507 Ki = 228 nM T67684 CR0K3N 16125508 Ki = 1132 nM T67684 CS51VQ 16125509 Ki = 13.4 nM T67684 CKBU51 16125529 Ki = 727 nM T67684 CA32GJ 16125531 Ki = 282 nM T67684 CX9FC1 16125533 Ki = 507 nM T67684 CJ92YT 16125535 Ki = 335 nM T67684 C1IC0F 16125541 Ki = 1.89 nM T67684 CPU2J5 16125565 Ki = 1056 nM T67684 CR78XQ 16125566 Ki = 13.8 nM T67684 C29GWL 16125567 Ki = 3.15 nM T67684 CV03SP 16125568 Ki = 16.5 nM T67684 C56TCH 16125570 Ki = 83.7 nM T67684 CXE2Y7 16125571 Ki = 8.8 nM T67684 C2AUB0 16125585 Ki = 6.7 nM T67684 C52IGT 16125587 Ki = 1.76 nM T67684 C8EH5G 16125589 Ki = 1.89 nM T67684 CFNB10 16125591 Ki = 9.11 nM T67684 CZ51NP 16125593 Ki = 541 nM T67684 CW3U7K 16125618 Ki = 25.8 nM T67684 C3AI6K 16125619 Ki = 7.6 nM T67684 CG4AD1 16125620 Ki = 2.37 nM T67684 CR8BD3 16125621 Ki = 7.9 nM T67684 C3D4MK 16125622 Ki = 2057 nM T67684 C18TFL 16125623 Ki = 418 nM T67684 CIN56P 16125640 Ki = 356 nM T67684 CB5MC6 16125642 Ki = 1.04 nM T67684 CPM1Z9 16125646 Ki = 1.84 nM T67684 C81PZO 16125648 Ki = 22.9 nM T67684 CFKE18 16125679 Ki = 53.5 nM T67684 C91FGA 16125680 Ki = 4.32 nM T67684 CMN0P3 16125681 Ki = 6.7 nM T67684 C4BYI2 16125682 Ki = 4.83 nM T67684 C1M2KX 16125683 Ki = 4.54 nM T67684 C91OQV 16125698 Ki = 2.61 nM T67684 CO02CS 16125704 Ki = 1.62 nM T67684 CA6PB8 16132042 Ki = 619 nM T67684 CZ2IS9 16660294 Ki > 10000 nM T67684 CEA26S 16664965 Ki = 0.75 nM T67684 CO1W8M 16721019 Ki = 2.1 nM T67684 CDB83R 17516658 EC50 > 30000 nM T67684 C7T8JC 19958494 Ki > 10000 nM T67684 C6LI5E 19958507 Ki > 10000 nM T67684 C3T5HF 21509921 Ki = 3761 nM T67684 CBN84K 22065997 Ki > 10000 nM T67684 C5WCD3 22745278 EC50 = 113 nM T67684 C3IQT5 23352279 Ki = 2600 nM T67684 C5SUY3 23352285 Ki = 4800 nM T67684 CXCO68 24192587 Ki = 384 nM T67684 C8KTP0 24739387 IC50 = 3000 nM T67684 C70CVK 24739554 IC50 > 10000 nM T67684 CSDA50 24739886 IC50 = 11000 nM T67684 C7I4LK 24750278 IC50 = 150 nM T67684 CVHL07 24758141 IC50 = 0.03162 nM T67684 C1V2UI 24764458 Ki = 0.73 nM T67684 CY21RE 24841480 Ki = 66 nM T67684 C4SY8G 24846938 Ki = 6.55 nM T67684 CF26NI 24865894 EC50 = 407.38 nM T67684 CI65LR 24876564 Ki = 0.765 nM T67684 C43RTZ 24882193 IC50 > 50000 nM T67684 C9YN3A 24894514 Ki = 52480.75 nM T67684 C8ND1U 24894515 Ki = 81283.05 nM T67684 CX2HR8 24894516 Ki = 33113.11 nM T67684 CG4B9R 24894624 Ki = 21379.62 nM T67684 C7KF9R 24894626 Ki = 2691.53 nM T67684 CFA60S 24894627 Ki = 2754.23 nM T67684 CT8B3K 24894629 Ki = 6918.31 nM T67684 CMF04K 24894631 Ki = 44668.36 nM T67684 CP08SJ 24894632 Ki = 22908.68 nM T67684 CLJK58 24894633 Ki = 28840.32 nM T67684 CR86FA 24894634 Ki = 17782.79 nM T67684 C9J3NX 24894636 Ki = 7762.47 nM T67684 CUY89J 24936155 Ki = 1200 nM T67684 CW4X0E 24962988 Ki = 635 nM T67684 CR7D1L 24967746 EC50 = 79.43 nM T67684 CK78XY 24988273 IC50 = 3.162 nM T67684 CD0OC3 24988641 IC50 = 1 nM T67684 CAY90E 24988642 IC50 = 2.512 nM T67684 COI7Y5 24988643 IC50 = 1.259 nM T67684 CYS4C3 24988644 IC50 = 0.2512 nM T67684 C4P3SV 24988645 IC50 = 0.1 nM T67684 CT93PZ 25010559 Ki = 0.3162 nM T67684 C5MYC3 25010776 EC50 > 30000 nM T67684 C1VRJ3 25014630 IC50 = 4500 nM T67684 C18VYH 25015647 EC50 > 40000 nM T67684 CA20NZ 25025581 Ki = 63.1 nM T67684 C8JW9U 25034110 IC50 = 3162.28 nM T67684 C9OC1I 25034111 IC50 = 15.85 nM T67684 C3DB4P 25034112 IC50 = 19952.62 nM T67684 CH67WY 25034180 IC50 = 1584.89 nM T67684 CBY3O2 25070582 IC50 = 300 nM T67684 CXBF68 25110764 EC50 > 50000 nM T67684 C50IKG 25110765 EC50 > 50000 nM T67684 CK0BT7 25147647 Ki > 10000 nM T67684 CE2OG1 25199525 EC50 > 15848.93 nM T67684 CRFJ43 25207745 EC50 = 3981.07 nM T67684 CP2T6G 25230693 EC50 = 630.96 nM T67684 C45ZNS 42596928 Ki = 3.631 nM T67684 C5DC7E 42598357 EC50 = 2511.89 nM T67684 CO6QB0 42598358 EC50 = 794.33 nM T67684 CDPA93 42598359 EC50 = 1258.93 nM T67684 CAM5P6 42598360 EC50 = 1584.89 nM T67684 C58SRK 42598586 EC50 = 398.11 nM T67684 CYL45Z 42598591 EC50 = 63.1 nM T67684 C6S2HI 42598828 EC50 = 1995.26 nM T67684 C2GYA4 42598829 EC50 = 1995.26 nM T67684 C5CZ7P 42599068 EC50 = 316.23 nM T67684 C7O2ZV 42599070 EC50 = 125.89 nM T67684 C6BUZ5 42599071 EC50 = 3162.28 nM T67684 C96IRU 42625858 IC50 = 2824000 nM T67684 C3IPM1 42625860 IC50 = 122000 nM T67684 C1KC8T 42625933 IC50 = 935000 nM T67684 CW09UI 42625935 IC50 = 1956000 nM T67684 CB7RF2 42625937 IC50 = 850000 nM T67684 C45KFN 42625939 IC50 = 29509000 nM T67684 CK54QN 42625941 IC50 = 829000 nM T67684 CIGB45 42625943 IC50 < 10000 nM T67684 CK31VL 42626010 IC50 = 306000 nM T67684 CZX8I4 42626012 IC50 < 10000 nM T67684 C5ME3B 42626014 IC50 = 5403000 nM T67684 C1KR9D 42626016 IC50 < 10000 nM T67684 CT62VZ 42626018 IC50 < 10000 nM T67684 CS74IR 42626087 IC50 = 22000 nM T67684 CED27C 42626089 IC50 < 10000 nM T67684 C7RF3J 42626091 IC50 = 13000 nM T67684 C42BZD 42626093 IC50 < 10000 nM T67684 C5THV8 42626095 IC50 = 36000 nM T67684 CF23ZA 42853213 Ki = 100 nM T67684 CQJ5Z1 42853214 Ki = 25.12 nM T67684 C3ABS1 44158142 EC50 = 2200 nM T67684 C2AV1K 44190762 IC50 = 1560 nM T67684 CMR7T1 44204999 EC50 > 25118.86 nM T67684 CPW7K9 44232679 IC50 = 0.37 nM T67684 CU2T6F 44232680 IC50 = 0.59 nM T67684 CEQO63 44232682 IC50 = 0.61 nM T67684 CW1V2M 44232684 IC50 = 0.48 nM T67684 C0J1FT 44232699 IC50 = 10 nM T67684 C2AX1T 44232701 IC50 = 11 nM T67684 C6M7JT 44232705 IC50 = 65 nM T67684 C34EAS 44232707 IC50 = 112 nM T67684 CZ38KJ 44232709 IC50 = 290 nM T67684 CDRG51 44232927 IC50 = 0.23 nM T67684 CVQB56 44232930 IC50 = 0.31 nM T67684 C4MK8P 44232931 IC50 = 0.39 nM T67684 CR05PU 44232946 IC50 = 17 nM T67684 C8GWI6 44232948 IC50 < 10 nM T67684 C0I6AD 44232950 IC50 = 23 nM T67684 CU6Q8I 44232952 Ki = 0.1585 nM T67684 C91ZIE 44232953 IC50 = 1939 nM T67684 C4OK7Y 44233172 IC50 = 1.04 nM T67684 C4Y3XC 44233174 IC50 = 1.04 nM T67684 CYC26A 44233176 IC50 = 0.24 nM T67684 C6WXJ9 44233187 IC50 = 1059 nM T67684 CJ97RM 44233188 IC50 < 10 nM T67684 CQM1T9 44233189 IC50 = 687 nM T67684 CAHP03 44233190 Ki = 2.512 nM T67684 CA59KP 44233191 Ki = 2.512 nM T67684 C8LM6H 44233399 Ki = 0.08 nM T67684 CCK0D4 44233400 IC50 = 0.24 nM T67684 C3OY7U 44233402 IC50 = 0.25 nM T67684 CP1G4K 44233417 IC50 = 1338 nM T67684 CA7LB8 44233419 IC50 = 2895 nM T67684 C5Q3EJ 44233675 IC50 = 206 nM T67684 CHK5U6 44233928 IC50 = 839 nM T67684 C5W7AP 44233929 IC50 < 10 nM T67684 C9OG5Z 44234194 IC50 = 2732 nM T67684 C5HA6K 44234429 IC50 > 10000 nM T67684 CET24J 44234431 IC50 = 25 nM T67684 CF4LQ7 44234680 IC50 = 74 nM T67684 CGL79K 44234682 IC50 = 37 nM T67684 CT87XH 44234685 IC50 = 65 nM T67684 CQF4S9 44234687 IC50 < 10 nM T67684 CQP25M 44234689 IC50 < 10 nM T67684 CX21NW 44235638 IC50 = 94 nM T67684 C17PIF 44235871 IC50 = 0.92 nM T67684 CBU6A0 44236098 IC50 = 0.42 nM T67684 CK0JC2 44236099 IC50 = 0.7 nM T67684 CUD0K2 44236100 IC50 = 0.28 nM T67684 CG13KU 44236331 IC50 = 0.71 nM T67684 CH12JO 44236333 IC50 = 0.96 nM T67684 C73FXN 44236335 IC50 = 0.6 nM T67684 CR8WZ1 44236337 IC50 = 200 nM T67684 CA15LQ 44236339 IC50 = 0.45 nM T67684 CF9TE1 44247935 Ki = 76 nM T67684 CGR6J0 44251556 EC50 > 30000 nM T67684 C2K0VZ 44253016 EC50 = 3981.07 nM T67684 C2LFH7 44274302 Ki = 14125.38 nM T67684 CZX4M3 44274317 Ki = 61659.5 nM T67684 C5L3FV 44274400 Ki = 40738.03 nM T67684 CF47ZS 44274417 Ki = 63095.73 nM T67684 CCK63Z 44274432 Ki = 72443.6 nM T67684 CZ1U0E 44274433 Ki = 45708.82 nM T67684 C3XP7C 44274441 Ki = 10000 nM T67684 CO1RL0 44274468 Ki = 27542.29 nM T67684 C9JX7D 44274469 Ki = 21379.62 nM T67684 CF36IC 44274477 Ki = 97723.72 nM T67684 CE20CZ 44275807 Ki = 1659.59 nM T67684 CC2OD4 44278111 Ki > 10000 nM T67684 CRMA84 44278114 Ki > 10000 nM T67684 CF0Y4M 44278115 Ki > 10000 nM T67684 C9Z0LT 44299564 Ki = 794.33 nM T67684 CX28HR 44299589 Ki = 676.08 nM T67684 CPL36O 44299599 Ki = 10964.78 nM T67684 CFN95A 44299616 Ki = 1949.84 nM T67684 CE4L1V 44299635 Ki = 5011.87 nM T67684 C9TWN3 44302727 IC50 = 10804.1 nM T67684 C5S8UL 44302728 IC50 = 1616.4 nM T67684 CQ4B5T 44302741 IC50 = 1482.3 nM T67684 C0AZF5 44302755 IC50 = 10315.1 nM T67684 CR5T1J 44302775 IC50 = 2629 nM T67684 CY8PD1 44302776 IC50 = 2720.9 nM T67684 C7GY5J 44302788 IC50 = 3394 nM T67684 CAV72D 44302793 IC50 = 32589.6 nM T67684 CV9QM6 44302813 IC50 = 5493.9 nM T67684 C43QTF 44302833 IC50 = 2827.7 nM T67684 CF74EQ 44302834 IC50 = 3067.8 nM T67684 C6J3EY 44302879 IC50 = 12612.2 nM T67684 CIU20B 44302900 IC50 = 2817 nM T67684 CGNA91 44302901 IC50 = 15293.8 nM T67684 C1RGS9 44304818 Ki = 18000 nM T67684 C03MFZ 44308733 Ki = 3.3 nM T67684 CT3V7Z 44308746 Ki = 8.3 nM T67684 C0Z3JQ 44308798 Ki = 2400 nM T67684 CN9M6A 44308799 Ki = 930 nM T67684 C38WIK 44308809 Ki = 100 nM T67684 CF06ON 44308818 Ki = 93 nM T67684 C90FZB 44308831 Ki = 120 nM T67684 CK14IH 44308832 Ki = 1.2 nM T67684 COE23J 44308861 Ki = 1.7 nM T67684 CMX10C 44308899 Ki = 1.1 nM T67684 CN5G8U 44308900 Ki = 9.6 nM T67684 CLJ71S 44308910 Ki = 50 nM T67684 C3L7HC 44308912 Ki = 2.9 nM T67684 CP0G8R 44308913 Ki = 16 nM T67684 CY6TU4 44309089 Ki = 17 nM T67684 CMAC70 44309090 Ki = 89 nM T67684 CND98T 44309107 Ki = 650 nM T67684 CEFY94 44309108 Ki = 290 nM T67684 C61LZX 44309135 Ki = 76 nM T67684 CY8D9F 44309151 Ki = 47 nM T67684 CD7QT6 44309153 Ki = 11 nM T67684 C7CQ3N 44309208 Ki = 17 nM T67684 C3B0IJ 44309209 Ki = 26 nM T67684 CIG89A 44309231 Ki = 7 nM T67684 CH7IJ2 44311760 Ki = 121.6 nM T67684 CT41MZ 44311762 Ki = 3.4 nM T67684 CT6Y9V 44311771 Ki = 10.1 nM T67684 CVX13Q 44318736 Ki = 450 nM T67684 CT58BQ 44318766 Ki = 7500 nM T67684 CLDG78 44318781 Ki = 794.33 nM T67684 CAH58Q 44318782 Ki = 0.7943 nM T67684 CR2T3J 44318817 Ki = 7400 nM T67684 C89JNT 44318928 Ki = 3.981 nM T67684 CL0HY5 44318929 Ki = 6700 nM T67684 C01CVA 44318930 Ki = 3000 nM T67684 C9Q6ET 44318969 Ki = 158.49 nM T67684 CZOA25 44319006 Ki = 25.12 nM T67684 CM0VD2 44319008 Ki = 158.49 nM T67684 CP9WF7 44319009 Ki = 1.585 nM T67684 C46OXB 44319010 Ki = 15.85 nM T67684 CT07JE 44319016 Ki = 25.12 nM T67684 CZ96OC 44319017 Ki = 31.62 nM T67684 C0C2XL 44319043 Ki = 3.981 nM T67684 C9SDP3 44319071 Ki = 1.259 nM T67684 C7R9DO 44319339 Ki = 2.512 nM T67684 C93POZ 44319342 Ki = 1.995 nM T67684 CGSU92 44326538 Ki = 243 nM T67684 CSE35C 44328347 Ki = 6900 nM T67684 CM6D4U 44328348 Ki > 5000 nM T67684 CX4M2I 44328356 Ki = 17000 nM T67684 C8O4PB 44328540 Ki = 1500 nM T67684 CTX68J 44328560 Ki >> 200 nM T67684 CP5W3M 44328561 Ki = 2000 nM T67684 CSK4B0 44346542 IC50 = 1308 nM T67684 CU2X1V 44356367 IC50 = 5400 nM T67684 CXJ4G7 44364174 Ki = 18 nM T67684 C3VT2M 44379080 Ki = 79.1 nM T67684 CU68GE 44379281 Ki = 39.2 nM T67684 CUA24S 44379508 Ki = 33.5 nM T67684 C7YTV9 44385809 Ki = 3.3 nM T67684 CHD9O7 44386115 Ki = 2.1 nM T67684 C1B4QL 44403095 Ki > 10000 nM T67684 C1YL7Z 44403098 Ki > 10000 nM T67684 CFV98A 44403101 Ki > 10000 nM T67684 C6OY9S 44403102 Ki > 10000 nM T67684 CH4SX6 44403105 Ki > 10000 nM T67684 C12FIH 44403106 Ki > 10000 nM T67684 C4LKC1 44404394 Ki > 10000 nM T67684 C3EJ4G 44404396 Ki > 10000 nM T67684 CT8S1N 44406268 Ki = 1 nM T67684 C43QUG 44406316 Ki = 2.5 nM T67684 C6B1HT 44406321 Ki = 7.9 nM T67684 CO14PG 44406342 Ki = 631 nM T67684 CPYG54 44406346 Ki = 40 nM T67684 CX7SG3 44406387 Ki = 100 nM T67684 C3G6PR 44406395 Ki = 7.9 nM T67684 C3UAN2 44406406 Ki = 4 nM T67684 C95QHZ 44406424 Ki = 1000 nM T67684 C6I3KL 44406451 Ki = 100 nM T67684 CX6L1E 44406476 Ki = 20 nM T67684 CMR10G 44406480 Ki = 10 nM T67684 C4SC6T 44406481 Ki = 0.4 nM T67684 C16NYM 44406520 Ki = 13 nM T67684 CVL24Q 44406521 Ki = 1.3 nM T67684 C3ZV2I 44406527 Ki = 50 nM T67684 CQCH24 44406572 Ki = 63 nM T67684 CRMB45 44406573 Ki = 0.2 nM T67684 CH5D2N 44406597 Ki = 0.25 nM T67684 C0A1PB 44406598 Ki = 1 nM T67684 CY0DB3 44406662 Ki = 0.32 nM T67684 CZM93T 44406686 Ki = 0.79 nM T67684 CZX87U 44406689 Ki = 7.9 nM T67684 CP0J2E 44406690 Ki = 1 nM T67684 C6GLV1 44408714 Ki = 2398.83 nM T67684 C6RFB5 44409461 Ki = 501 nM T67684 C8H5WF 44409462 Ki = 100 nM T67684 CX7R9U 44409463 Ki = 50 nM T67684 C1JN2W 44409556 Ki = 501 nM T67684 C48TAF 44409557 Ki = 3200 nM T67684 CL1UM2 44409558 Ki = 13 nM T67684 C65LDN 44409651 Ki = 50 nM T67684 C41BTQ 44409653 Ki = 32 nM T67684 C7UE8I 44409654 Ki = 158 nM T67684 CR5N4B 44409660 Ki = 790 nM T67684 CTH4U7 44409744 Ki = 251 nM T67684 C1SNK8 44409745 Ki = 63 nM T67684 C1DR6L 44409746 Ki = 251 nM T67684 CU5PZ9 44409749 Ki = 316 nM T67684 CLWK34 44409751 Ki = 7.9 nM T67684 CVUL24 44409754 Ki = 79 nM T67684 CXQ1E6 44409755 Ki = 100 nM T67684 CSK9M0 44409759 Ki = 16 nM T67684 COZ39R 44409760 Ki = 316 nM T67684 C58LXG 44409765 Ki = 32 nM T67684 C5Y9MU 44409769 Ki = 398 nM T67684 CQI9A1 44409772 Ki = 100 nM T67684 CNJC24 44409787 Ki = 2512 nM T67684 CN06AV 44409796 Ki = 398 nM T67684 CU4KQ2 44409797 Ki = 200 nM T67684 CWPZ82 44409937 Ki = 79 nM T67684 CS6UR7 44409944 Ki = 10 nM T67684 C5VFP3 44409945 Ki = 7.9 nM T67684 CBXV64 44409956 Ki = 25 nM T67684 CUV53S 44409961 Ki = 126 nM T67684 C4XBR6 44409962 Ki = 316 nM T67684 C4VZ5R 44409963 Ki = 501 nM T67684 CU64VF 44409965 Ki = 398 nM T67684 CAR61H 44409976 Ki = 63 nM T67684 CLT2Y3 44409977 Ki = 126 nM T67684 C48QIT 44409978 Ki = 79 nM T67684 CK46WN 44409981 Ki = 40 nM T67684 CY0F6E 44409982 Ki = 79 nM T67684 C4QTI3 44415886 Ki = 2.4 nM T67684 CC9AV3 44418764 Ki = 316.23 nM T67684 CV6UQ3 44419370 Ki > 100000 nM T67684 CH85PD 44420788 Ki = 2535 nM T67684 C84KBW 44420791 Ki = 153 nM T67684 C2P7XQ 44420794 Ki = 0.67 nM T67684 CS9XH3 44420821 Ki = 4.1 nM T67684 C2N5LX 44422691 EC50 = 275.42 nM T67684 CIRB78 44422696 Ki = 23442.29 nM T67684 CHT24X 44422698 Ki = 36307.81 nM T67684 CDE8A1 44428745 Ki = 213.8 nM T67684 CJT90I 44430454 Ki = 1.3 nM T67684 CD8Z6V 44430456 Ki = 79 nM T67684 CQJA76 44430457 Ki = 40 nM T67684 C8KO4X 44430461 Ki = 32 nM T67684 CEL85Z 44430462 Ki = 158 nM T67684 C1WA3Q 44430464 Ki = 200 nM T67684 C7L8CO 44430466 Ki = 794 nM T67684 CJ6Z8U 44430467 Ki = 158.49 nM T67684 CL0VG4 44430469 Ki = 631 nM T67684 C9SQ4Y 44430470 Ki = 40 nM T67684 CFRQ71 44430472 Ki = 79 nM T67684 CYQ0N1 44430473 Ki = 13 nM T67684 CQIA96 44430474 Ki = 501 nM T67684 CRN6M1 44431367 Ki = 20 nM T67684 CQD71K 44431369 Ki = 18 nM T67684 CAE86V 44431370 Ki = 20 nM T67684 C92HNF 44431372 Ki = 56 nM T67684 CR5U1K 44431374 IC50 > 100 nM T67684 CI36TZ 44431375 Ki = 23 nM T67684 CZ12VG 44431376 Ki = 19 nM T67684 CV5LX1 44431377 IC50 > 100 nM T67684 CHI3W5 44431378 IC50 > 100 nM T67684 C6X2EZ 44431379 IC50 > 100 nM T67684 CS0H4C 44431380 Ki = 4.9 nM T67684 C5FJR6 44431381 Ki = 3.3 nM T67684 CG0BM9 44431382 Ki = 2.5 nM T67684 CW60PY 44431383 Ki = 2.7 nM T67684 C0JL9K 44431384 Ki = 1.5 nM T67684 C3S0AU 44431386 Ki = 14 nM T67684 C0T5AL 44431387 Ki = 6.8 nM T67684 C15WZI 44431388 Ki = 5.8 nM T67684 C29VWS 44431389 Ki = 2.9 nM T67684 C1LJ6G 44431391 Ki = 4.2 nM T67684 CLA76R 44431393 Ki = 0.22 nM T67684 C9TN6X 44431394 IC50 > 100 nM T67684 COX18J 44431395 IC50 > 100 nM T67684 CG45PO 44437242 Ki = 3995 nM T67684 C6I2JO 44437248 Ki = 7386 nM T67684 CZI05O 44437258 Ki = 1448 nM T67684 C7VP1Y 44437297 Ki = 4740 nM T67684 C5GT7C 44437302 Ki = 5539 nM T67684 C37QFT 44437307 Ki = 887 nM T67684 C36LXN 44446840 Ki = 35481.34 nM T67684 CVT7J2 44449463 Ki = 2.512 nM T67684 C12XGE 44456400 Ki > 10000 nM T67684 C4DL5C 44469677 IC50 > 10000 nM T67684 C7Y3RF 44552684 IC50 = 0.1259 nM T67684 C1E3MT 44554514 Ki = 3.7 nM T67684 CVA67X 44568347 Ki = 170 nM T67684 CY9C2A 44571572 Ki > 100000 nM T67684 CGJW09 44573263 IC50 = 1258.93 nM T67684 C4TZ6Y 44573264 IC50 = 199.53 nM T67684 C4CXZ3 44573265 IC50 = 316.23 nM T67684 C5IAC6 44573370 IC50 = 251.19 nM T67684 CJ3D7W 44573371 IC50 = 3162.28 nM T67684 CHG7Y1 44573372 IC50 = 2511.89 nM T67684 CGJ47U 44573373 IC50 > 10000 nM T67684 CPVC16 44573420 IC50 = 251.19 nM T67684 C3J8IY 44573421 IC50 = 6309.57 nM T67684 C6RZ9M 44573422 IC50 = 7943.28 nM T67684 CM18WY 44573423 IC50 = 316.23 nM T67684 C5PL0E 44573465 IC50 = 79.43 nM T67684 C3FPY5 44573466 IC50 = 501.19 nM T67684 CI5BF3 44573499 IC50 = 501.19 nM T67684 CWEJ21 44573500 IC50 = 1000 nM T67684 CVYZ93 44573501 IC50 = 316.23 nM T67684 C2B6XS 44573543 IC50 = 3981.07 nM T67684 CC9D0M 44573544 IC50 = 630.96 nM T67684 CY75PH 44573545 IC50 = 794.33 nM T67684 C5BU9J 44573578 IC50 = 19.95 nM T67684 C1N5XD 44573619 IC50 = 199.53 nM T67684 C1ETX5 44573620 IC50 = 501.19 nM T67684 CK9GC6 44573621 IC50 = 1258.93 nM T67684 CI4H9J 44573661 IC50 = 1995.26 nM T67684 CJ60ZS 44573662 IC50 = 251.19 nM T67684 CNRU68 44573663 IC50 = 316.23 nM T67684 CD3V6E 44573744 IC50 = 1584.89 nM T67684 C10RJW 44573745 IC50 = 6309.57 nM T67684 C9PVC8 44573746 IC50 > 10000 nM T67684 CD0KL6 44573785 IC50 = 630.96 nM T67684 CWTN35 44573786 IC50 = 5011.87 nM T67684 COV92W 44573787 IC50 > 10000 nM T67684 CN68YI 44578707 Ki > 10000 nM T67684 CHUN40 44578928 EC50 > 50000 nM T67684 CZYP06 44578975 EC50 > 50000 nM T67684 CCIT12 44578976 EC50 > 50000 nM T67684 CW53ZF 44578977 EC50 > 50000 nM T67684 CYHM34 44578978 EC50 > 50000 nM T67684 CGF7A4 44579375 EC50 > 50000 nM T67684 C1OCB6 44579416 EC50 > 50000 nM T67684 CARW17 44579417 EC50 > 50000 nM T67684 C2DFV7 44579418 EC50 > 50000 nM T67684 CTC8H6 44579419 EC50 > 50000 nM T67684 CYR0O3 44579457 EC50 > 50000 nM T67684 CF1EA4 44579458 EC50 > 50000 nM T67684 C6HMP4 44589495 IC50 = 10 nM T67684 C9U3KY 44589496 IC50 = 5.012 nM T67684 CXL82E 44589497 IC50 = 251.19 nM T67684 CLGW57 44589498 IC50 = 100 nM T67684 C1KY5I 44589499 IC50 = 2511.89 nM T67684 C0N4QF 44589529 IC50 = 316.23 nM T67684 CQ4Y8O 44589531 EC50 > 30000 nM T67684 COE0T7 44589569 IC50 = 501.19 nM T67684 CE4FX5 44589570 IC50 = 100 nM T67684 C9J2RO 44589571 IC50 = 158.49 nM T67684 CKY4F8 44589572 IC50 = 501.19 nM T67684 CX19BO 44589573 IC50 = 1584.89 nM T67684 C10LXB 44589574 IC50 = 398.11 nM T67684 CUD4M8 44589575 IC50 = 1000 nM T67684 CL40CM 44589593 EC50 > 30000 nM T67684 CKS5V4 44589594 EC50 > 30000 nM T67684 CXB30W 44589595 EC50 > 30000 nM T67684 CM5LJ8 44589596 EC50 > 30000 nM T67684 CPXE19 44589643 EC50 > 30000 nM T67684 C8AJO6 44589644 EC50 > 30000 nM T67684 CFS1A4 44589645 EC50 > 30000 nM T67684 C71EHI 44589646 EC50 > 30000 nM T67684 CQB5A9 44589681 EC50 = 113 nM T67684 CE06LX 44589984 IC50 = 19.95 nM T67684 C6LC7V 44590033 IC50 = 19.95 nM T67684 CL57OY 44590034 IC50 = 25.12 nM T67684 CO3GX2 44590035 IC50 = 50.12 nM T67684 CT58OX 44590036 IC50 = 31.62 nM T67684 C2H9IW 44590122 IC50 = 6.31 nM T67684 CJ2M0R 44590123 IC50 = 7.943 nM T67684 C5JVF6 44590124 IC50 = 15.85 nM T67684 C3G5LY 44590125 IC50 = 15.85 nM T67684 CF4DI1 44590166 IC50 = 794.33 nM T67684 CYC47W 44590167 IC50 = 25.12 nM T67684 CH61KJ 44590182 IC50 = 25.12 nM T67684 CUA62X 44593616 Ki = 281.84 nM T67684 CN9ID8 44593617 Ki = 302 nM T67684 CDM56I 44593618 Ki = 42.66 nM T67684 CU63PQ 44593619 Ki = 18.2 nM T67684 CL8D2S 44593620 Ki = 23.99 nM T67684 CI97KQ 44593621 Ki = 346.74 nM T67684 CNZ1U7 44593651 IC50 < 1 nM T67684 CL5O8E 44602489 EC50 > 30000 nM T67684 C5KTS1 44609903 Ki = 3.7 nM T67684 CH2Z3O 44610056 Ki = 0.29 nM T67684 C9G8WB 44610361 Ki = 18 nM T67684 CO3I5F 44622849 Ki = 8200 nM T67684 CVZ6Y1 44627739 Ki = 95.5 nM T67684 CE6A9F 44627740 Ki = 7.762 nM T67684 C6EU7P 44627741 Ki = 85.11 nM T67684 CW40TR 44627742 Ki = 33.88 nM T67684 C5GIU6 44627743 Ki = 36.31 nM T67684 CK9DO1 44627745 Ki = 7.244 nM T67684 CJ8S1L 44627747 Ki = 23.44 nM T67684 C5LY8C 44627851 Ki = 8.913 nM T67684 CC4A3X 44627853 Ki = 1.66 nM T67684 CH4N5J 44627854 Ki = 23.44 nM T67684 CO8C6D 44627855 Ki = 323.59 nM T67684 COL8E1 44627856 Ki = 1659.59 nM T67684 C6WS7M 44627857 Ki = 1.514 nM T67684 C43BJY 44627859 Ki = 9.333 nM T67684 CW0X6A 44627955 Ki = 154.88 nM T67684 CXNF31 44627957 Ki = 512.86 nM T67684 C4LOY2 45115589 Ki < 1000 nM T67684 C9U0VH 45259185 Ki = 263.03 nM T67684 CNC1R2 45259186 Ki = 51.29 nM T67684 CP2CZ7 45259187 Ki = 288.4 nM T67684 CW14TS 45259188 Ki = 4.169 nM T67684 CO8W1X 45259189 Ki = 6.918 nM T67684 CF16YZ 45259190 Ki = 77.62 nM T67684 C1K0ZH 45259193 Ki = 31.62 nM T67684 C7L1CU 45266348 Ki = 34.67 nM T67684 CJQ8C6 45266387 IC50 = 15.85 nM T67684 C2IV6N 45266389 IC50 = 12.59 nM T67684 C7WBU9 45266390 IC50 = 15.85 nM T67684 C5J2TE 45266397 IC50 = 6.31 nM T67684 C0O9TA 45266401 IC50 = 25.12 nM T67684 C5P1NR 45266404 IC50 = 125.89 nM T67684 CJ9W5C 45266406 IC50 = 6.31 nM T67684 CH74XR 45266408 IC50 = 7.943 nM T67684 CGH8T0 45266411 IC50 = 1258.93 nM T67684 C73TVO 45266437 IC50 = 15.85 nM T67684 C9IHS7 45266451 IC50 = 2511.89 nM T67684 C7JR0B 45266454 IC50 > 10000 nM T67684 C5PTZ9 45266459 IC50 = 39.81 nM T67684 C0D4LK 45266462 IC50 = 15.85 nM T67684 CUK8N1 45266464 IC50 = 50.12 nM T67684 CRI98L 45266467 IC50 = 6.31 nM T67684 C0AV6F 45266469 IC50 = 1.995 nM T67684 CZA73U 45266470 IC50 = 12.59 nM T67684 C0FHW1 45266476 IC50 = 31.62 nM T67684 CZ23VF 45266478 IC50 = 10 nM T67684 CK6X3B 45786849 Ki = 10000 nM T67684 CL0M1G 46174144 Ki = 0.06 nM T67684 CU4V5R 46227410 Ki = 44668.36 nM T67684 CWQ1L9 46227412 Ki = 10964.78 nM T67684 CX2E6A 46227414 Ki > 100000 nM T67684 C0Z4RD 46227416 Ki > 100000 nM T67684 CK2R5G 46227454 Ki > 100000 nM T67684 C8OZI6 46227456 Ki = 21379.62 nM T67684 CB45NM 46227458 Ki = 77624.71 nM T67684 C1J0IF 46227460 Ki = 32359.37 nM T67684 CQ4DI6 46227480 Ki = 46773.51 nM T67684 CHKL80 46227482 Ki = 16218.1 nM T67684 CVP7T6 46227484 Ki = 10471.29 nM T67684 CC6RH5 46227486 Ki = 40738.03 nM T67684 CSQ0V3 46227554 Ki = 66069.34 nM T67684 CK1X9S 46830361 IC50 = 3700 nM T67684 C1Q0MH 46830362 IC50 = 4200 nM T67684 CH3ID7 46830363 IC50 > 10000 nM T67684 CH83EL 46854806 Ki = 550 nM T67684 C01YTE 46871665 IC50 = 1000 nM T67684 CUY51M 46871666 IC50 = 1258.93 nM T67684 CYLZ50 46871844 IC50 = 39.81 nM T67684 CK8A1O 46880462 Ki > 10000 nM T67684 C9KDP4 46880463 Ki > 10000 nM T67684 CODR73 46880498 Ki > 10000 nM T67684 CHJ5Y6 46880566 Ki > 10000 nM T67684 CE9PG2 46880567 Ki > 10000 nM T67684 C01PGO 46880568 Ki > 10000 nM T67684 CS7L4X 46880569 Ki > 10000 nM T67684 C0PXY7 46880628 Ki > 10000 nM T67684 CD37LU 46880629 Ki > 10000 nM T67684 CUY89F 46880630 Ki > 10000 nM T67684 C4P6XS 46880631 Ki > 10000 nM T67684 CJ53KF 46880672 Ki > 10000 nM T67684 CYJC08 46880673 Ki > 10000 nM T67684 C1RI9O 46880674 Ki > 10000 nM T67684 CCZ5I8 46883796 IC50 = 4300 nM T67684 CVCF68 46883843 IC50 > 10000 nM T67684 C30KJT 46890906 IC50 = 1.995 nM T67684 CMCH59 46890907 IC50 = 12.59 nM T67684 CJ57WZ 46890960 IC50 = 1995.26 nM T67684 CD1MS4 46890962 IC50 = 125.89 nM T67684 C8QZ2Y 46890963 IC50 = 70 nM T67684 CW70YU 46890977 IC50 = 251.19 nM T67684 C0KDX8 46891020 IC50 = 19.95 nM T67684 CJ10MI 46891021 IC50 = 3981.07 nM T67684 CM01DZ 46891022 IC50 = 1258.93 nM T67684 CZ1EO8 46891075 IC50 = 2511.89 nM T67684 CJ74AZ 46891076 IC50 = 3162.28 nM T67684 CI9J3P 46891141 IC50 = 10000 nM T67684 C6P5JG 46891142 IC50 = 10000 nM T67684 C6I8NE 46891143 IC50 = 10000 nM T67684 CW03QZ 46891144 IC50 = 1258.93 nM T67684 CTSZ49 46891179 IC50 = 5011.87 nM T67684 COT8S4 46891375 EC50 > 10000 nM T67684 CW1YX7 46891488 IC50 = 3981.07 nM T67684 CB1Z5A 46905390 IC50 = 457.8 nM T67684 C67XQI 46945663 EC50 > 30000 nM T67684 C7IAW9 49663949 IC50 < 1500 nM T67684 C2LZJ0 49783209 Ki = 823 nM T67684 C57SMG 49783415 Ki = 1095 nM T67684 C0TG6I 49783419 Ki > 10000 nM T67684 C20SCO 49797320 Ki = 4013 nM T67684 C29QSB 49797322 Ki = 537 nM T67684 CT4QU7 49797325 Ki = 3919 nM T67684 CC7JK8 49797556 IC50 = 6599000 nM T67684 CX7YI2 49797557 IC50 = 1068000 nM T67684 C6WJ9C 49797558 IC50 = 145000 nM T67684 CPI6N0 49853777 IC50 > 100000 nM T67684 C94GDK 49853778 IC50 > 100000 nM T67684 CHV3U8 49853881 IC50 > 100000 nM T67684 CTBY97 49853883 IC50 > 100000 nM T67684 CQP63D 49853884 IC50 = 57000 nM T67684 CY8M9A 49853885 IC50 > 100000 nM T67684 CN0JU9 49853987 IC50 > 100000 nM T67684 C8DVX6 49855131 IC50 > 100000 nM T67684 C2RY0J 50878551 Ki > 10000 nM T67684 C1W6TV 50898777 Ki > 10000 nM T67684 CXMZ73 50898778 Ki > 10000 nM T67684 C3BZ7G 50925541 IC50 = 10 nM T67684 C7NGS9 50925542 IC50 = 1.259 nM T67684 CHG0K5 50925543 IC50 = 7.943 nM T67684 CE4KP1 51050257 Ki > 10000 nM T67684 CM47HJ 52176747 IC50 = 7000 nM T67684 CT16AY 52942401 IC50 = 19.95 nM T67684 CY6UC5 52942402 IC50 = 5.012 nM T67684 CLXF87 52942447 IC50 > 1000 nM T67684 CYQF74 52942458 IC50 = 100 nM T67684 CM3IV9 52942497 IC50 > 1000 nM T67684 C1G7HW 52942610 IC50 = 251.19 nM T67684 CZ3X0R 52942628 IC50 = 63.1 nM T67684 CE71SW 52942930 IC50 > 1000 nM T67684 CXT1M9 52943696 IC50 = 125.89 nM T67684 CZ78UX 52943721 IC50 = 316.23 nM T67684 C5O4MA 52943879 IC50 = 50.12 nM T67684 C5UN3Y 52943921 IC50 = 398.11 nM T67684 CFLA17 52944764 IC50 > 1000 nM T67684 CE04VX 52945165 IC50 = 398.11 nM T67684 CBTM43 52945272 IC50 = 3.981 nM T67684 CW49GK 52946068 IC50 = 398.11 nM T67684 C6YBT4 52946249 IC50 = 63.1 nM T67684 CJ85YX 52946359 IC50 = 199.53 nM T67684 CZT9U3 52947254 IC50 = 15.85 nM T67684 COW8Z9 52947320 IC50 = 100 nM T67684 CV81IX 52947552 IC50 = 100 nM T67684 CC4A1H 52947553 IC50 = 125.89 nM T67684 CF08DE 52948443 IC50 = 15.85 nM T67684 CBQ7X1 52949760 IC50 > 1000 nM T67684 CN91QX 52949883 IC50 = 794.33 nM T67684 CN0U6H 52949961 IC50 = 31.62 nM T67684 C2LEQ0 52950036 IC50 = 158.49 nM T67684 CR3XD8 53239456 Ki = 0.305 nM T67684 C6KU3Z 53303986 IC50 > 10000 nM T67684 CD0BK2 53317169 Ki = 77 nM T67684 C5OB4K 53317170 Ki = 0.53 nM T67684 C1PY6E 53318454 Ki = 22 nM T67684 CX1G3F 53318455 Ki = 28 nM T67684 CEH3U9 53319786 Ki = 50 nM T67684 C63GQX 53319787 Ki = 2.5 nM T67684 C3S1ZO 53319788 Ki = 32 nM T67684 CX85DT 53321084 Ki = 17 nM T67684 CP6M8S 53321085 Ki = 14 nM T67684 C7F6KA 53321086 Ki = 5.1 nM T67684 CTM5V2 53322411 Ki = 4.8 nM T67684 CUC51K 53322412 Ki = 7 nM T67684 C4CT2P 53323772 Ki = 0.75 nM T67684 CR4W9L 53324553 Ki = 1395 nM T67684 CFG0N5 53325043 Ki = 48 nM T67684 C54WXB 53325044 Ki = 84 nM T67684 CF96WZ 53325045 Ki = 1.8 nM T67684 CZ49NP 53325336 Ki = 67 nM T67684 CSQ08F 53325550 Ki = 19 nM T67684 CE16ZW 53326338 Ki = 55 nM T67684 CL29ZP 53326339 Ki = 25 nM T67684 CNAL81 53326340 Ki = 2.6 nM T67684 C58HUX 53326588 Ki = 1.6 nM T67684 CNS26Q 53326837 Ki = 4.6 nM T67684 CT1BP8 53326849 Ki = 98 nM T67684 CMX05A 53326934 Ki = 9.5 nM T67684 CS1OI7 53382523 EC50 > 30000 nM T67684 CWR16G 53382542 EC50 > 30000 nM T67684 C7YP3A 53385782 EC50 > 10000 nM T67684 C6A7VE 53414666 Ki = 36000 nM T67684 C3KRU5 54580128 Ki = 0.091 nM T67684 CFNI73 54580129 Ki = 0.276 nM T67684 CF6X0Z 54580133 Ki = 4.7 nM T67684 C6D3OU 54580864 IC50 = 0.6 nM T67684 CM9KH3 54581928 IC50 = 19 nM T67684 CN03FM 54582151 Ki = 0.99 nM T67684 C1ZMV9 54582844 IC50 = 1.2 nM T67684 CA74TP 54583092 Ki = 0.397 nM T67684 C50PTV 54583100 Ki = 0.634 nM T67684 CMRC75 54583839 IC50 = 71.1 nM T67684 CZ82MJ 54583840 IC50 = 1.4 nM T67684 C01VQF 54584800 IC50 = 22.5 nM T67684 CHP9F8 54585742 IC50 = 796.8 nM T67684 CO5H6T 54585743 IC50 = 2.4 nM T67684 CB5IF2 54586723 IC50 = 659.3 nM T67684 CKTW24 54586742 IC50 = 18.6 nM T67684 CWXP12 54586744 IC50 = 0.9 nM T67684 CJC2E3 54586985 Ki = 6.1 nM T67684 C2ZYD7 54586986 Ki = 1.45 nM T67684 C2IJF0 54591014 IC50 = 1.585 nM T67684 CK01PH 54757332 Ki = 1.9 nM T67684 C0CLP1 54757541 Ki = 0.16 nM T67684 CVI3F5 54757542 Ki = 2 nM T67684 C85DPY 54757543 Ki = 0.76 nM T67684 CB02HA 54757544 Ki = 0.56 nM T67684 CUSR42 54757560 Ki = 10 nM T67684 CB8Y4V 54757653 Ki = 11 nM T67684 CYB78R 54757668 Ki = 2.5 nM T67684 CE1PR6 54757766 Ki = 7.3 nM T67684 CWYX94 54757772 Ki = 2.2 nM T67684 C6N1TA 54757856 Ki = 0.18 nM T67684 C8WHT5 56593934 Ki = 10000 nM T67684 CA9T3J 56667295 Ki = 0.88 nM T67684 CB0P9N 56944383 Ki > 1000 nM T67684 C1TC7Q 56963799 Ki = 512 nM T67684 C3WC7Z 56965018 Ki = 2.188 nM T67684 CUP4Y0 57326139 Ki = 17782.79 nM T67684 C1G9XY 57326141 Ki = 81283.05 nM T67684 CG3YS9 57326143 Ki = 9772.37 nM T67684 CCYU25 57326145 Ki = 31622.78 nM T67684 CS86GL 57326232 Ki = 61.66 nM T67684 C3AF0Z 57326234 Ki = 1.479 nM T67684 CLSW35 57326236 Ki = 8912.51 nM T67684 CL3R5D 57326238 Ki = 21379.62 nM T67684 C4G1LB 57326325 Ki = 72.44 nM T67684 C6CB9J 57326326 Ki = 1.514 nM T67684 CI4VR1 57390664 IC50 < 0.03162 nM T67684 CTO37G 57390665 IC50 = 0.07943 nM T67684 CD8A2S 57390666 IC50 = 0.3981 nM T67684 CT1ZM6 57390714 IC50 = 1 nM T67684 CVLF26 57390720 IC50 = 0.1585 nM T67684 CJ6BU8 57390766 IC50 = 0.1995 nM T67684 C5OJP0 57391102 EC50 > 30000 nM T67684 C7E2MF 57391636 IC50 = 0.1 nM T67684 C71CIS 57391772 IC50 = 158.49 nM T67684 CLO46H 57391773 IC50 = 0.631 nM T67684 CF6V2G 57391774 IC50 < 0.05012 nM T67684 CCW6F2 57391775 IC50 = 0.1259 nM T67684 CJVQ39 57392462 IC50 = 0.2512 nM T67684 C62MET 57392514 IC50 = 5.012 nM T67684 C4AEU8 57392515 IC50 = 0.5012 nM T67684 C2OPN7 57392520 IC50 = 0.1995 nM T67684 CS6DM5 57392521 IC50 = 0.1995 nM T67684 CUD91Z 57392578 IC50 = 0.05012 nM T67684 C17GMJ 57393065 IC50 > 30000 nM T67684 CMHO80 57393498 IC50 = 1.585 nM T67684 C9G3QD 57393500 IC50 = 10 nM T67684 CKLP94 57393501 IC50 = 5.012 nM T67684 CFW0R7 57393502 IC50 = 7.943 nM T67684 CD79JL 57393503 IC50 < 0.1 nM T67684 C41CLN 57394170 IC50 = 0.0631 nM T67684 CQZW06 57394233 IC50 = 0.3162 nM T67684 C6D2LP 57394234 IC50 = 0.0631 nM T67684 CT3R1F 57395096 IC50 = 0.1995 nM T67684 C9J2IX 57395097 IC50 = 0.3162 nM T67684 C6RIA9 57395222 IC50 = 0.05012 nM T67684 C1IC8Q 57395952 IC50 = 0.1585 nM T67684 CJ6H9D 57395989 IC50 = 0.631 nM T67684 CM34WX 57395990 IC50 = 0.07943 nM T67684 C1AYF4 57395991 IC50 = 0.1 nM T67684 CMWY05 57395997 IC50 = 1 nM T67684 CFIY54 57396059 IC50 < 0.0631 nM T67684 CJ49EH 57396866 IC50 = 0.3981 nM T67684 C8JK6R 57397002 IC50 = 0.7943 nM T67684 C2N0YJ 57397003 IC50 = 3.162 nM T67684 CDN31Q 57397742 IC50 = 6.31 nM T67684 CKG72A 57397743 IC50 = 1.585 nM T67684 C4ZRD7 57397744 IC50 = 0.1585 nM T67684 CSTF91 57397745 IC50 = 3.162 nM T67684 CQR81W 57397746 IC50 = 0.3162 nM T67684 CFJV31 57397747 IC50 = 3.162 nM T67684 C3ZQN0 57397790 IC50 = 1.259 nM T67684 C8BMT6 57397791 IC50 = 0.7943 nM T67684 C3RCW4 57397792 IC50 = 0.1259 nM T67684 CAX69Q 57397793 IC50 = 0.1995 nM T67684 CS9A5D 57397794 IC50 = 0.1995 nM T67684 C9C0ZE 57398751 IC50 = 0.1585 nM T67684 C27EQL 57399404 IC50 < 0.05012 nM T67684 CFE4A5 57399405 IC50 = 2.512 nM T67684 C9SMX1 57399406 IC50 = 0.3162 nM T67684 C64PHW 57399407 IC50 = 0.1995 nM T67684 C0E8MI 57399408 IC50 = 0.631 nM T67684 CTO46R 57400155 IC50 = 3.162 nM T67684 CCN82P 57400294 IC50 = 0.2512 nM T67684 CZ54JA 57400421 IC50 = 0.03162 nM T67684 CVM6H8 57400423 IC50 = 5.012 nM T67684 C62EVX 57400424 IC50 < 0.03981 nM T67684 CUVX70 57401170 IC50 = 1.259 nM T67684 C34UER 57401217 IC50 = 0.1995 nM T67684 C6GSH4 57401218 IC50 = 0.1995 nM T67684 C87UKH 57401219 IC50 = 0.1259 nM T67684 CNG85V 57401272 IC50 < 0.03981 nM T67684 CW5K7F 57401273 IC50 = 0.0631 nM T67684 CC7X9S 57402222 IC50 = 0.7943 nM T67684 CVL64H 57402223 IC50 = 251.19 nM T67684 CHD56A 57402931 IC50 = 0.1995 nM T67684 CNT75F 57402970 IC50 = 1.259 nM T67684 CS1W0Q 57403021 IC50 < 0.03162 nM T67684 CYZQ72 57403853 IC50 = 0.1585 nM T67684 C57FRE 57403964 IC50 = 1 nM T67684 C9OPD7 57403965 IC50 = 5.012 nM T67684 CC3B8P 57403966 IC50 < 0.05012 nM T67684 CQ5BG6 57525860 EC50 > 30000 nM T67684 C9TMZ3 57558000 Ki > 100000 nM T67684 CPV56A 58348375 IC50 = 0.07943 nM T67684 CA14SG 58653718 Ki > 100000 nM T67684 C2XDJ0 58975257 IC50 = 6399 nM T67684 C45JFO 59145957 Ki = 7.7 nM T67684 CKV58R 59179619 IC50 = 0.0631 nM T67684 C3WS7G 59707188 Ki = 1.1 nM T67684 CGO41Y 59707195 Ki = 5 nM T67684 CZ4CH7 60150385 IC50 = 85.2 nM T67684 CAZ9B3 62705488 IC50 > 10000 nM T67684 C9F4JW 62705832 IC50 > 10000 nM T67684 C3XL7O 66561967 Ki = 661 nM T67684 CZ0QX9 66604761 IC50 < 10 nM T67684 C9A8WH 66875589 Ki = 1.995 nM T67684 CB06GE 67547652 IC50 = 172.5 nM T67684 CDH6V7 67547661 IC50 = 130.5 nM T67684 CE91TN 67547949 IC50 = 64.4 nM T67684 CMA5W7 67548135 IC50 = 0.7 nM T67684 C8OC2K 67548543 IC50 = 60.2 nM T67684 CD41JS 67548925 IC50 = 0.7 nM T67684 C8MU9E 67549179 IC50 = 18.7 nM T67684 C9TAI0 68858512 IC50 < 10 nM T67684 C4I2WU 68859713 IC50 < 10 nM T67684 C1HJZ4 68859717 IC50 = 64 nM T67684 C8NE2T 68859719 IC50 < 10 nM T67684 C5WSY4 68859731 IC50 < 10 nM T67684 CSZH87 68860056 IC50 = 109 nM T67684 CBZ8A4 68860242 IC50 < 10 nM T67684 C1L9SF 68860730 IC50 < 10 nM T67684 C9P1TC 68860783 IC50 < 10 nM T67684 CFS4A0 68861304 IC50 < 10 nM T67684 CTW10U 69058945 Ki = 3.162 nM T67684 CQO63X 69167248 IC50 = 0.2512 nM T67684 C6TI9M 69444105 IC50 = 20.3 nM T67684 CF8DC9 70681307 Ki = 40.74 nM T67684 CUV5Y9 70681419 IC50 < 10 nM T67684 CXT67P 70683405 Ki = 39.81 nM T67684 CN98LU 70685504 Ki = 48.98 nM T67684 C4LJZ3 70685519 IC50 < 10 nM T67684 CT41UM 70687661 Ki = 44.67 nM T67684 CQ2VB3 70689728 IC50 < 10 nM T67684 C2R4HT 70691874 IC50 < 10 nM T67684 CI0V8T 70693915 IC50 < 10 nM T67684 CJLS94 71449148 Ki = 37.04 nM T67684 C9VZ8J 71450550 Ki = 543 nM T67684 C4M1WQ 71450615 IC50 = 223.2 nM T67684 C29VNS 71450616 IC50 = 6.1 nM T67684 CDN70A 71450617 IC50 = 237 nM T67684 C8HR1L 71450662 IC50 = 417.1 nM T67684 CY3M8B 71451570 IC50 > 1500 nM T67684 C4NDR3 71452382 Ki = 407 nM T67684 CYK20Z 71452384 Ki = 209 nM T67684 CDTW09 71452387 Ki = 1609 nM T67684 C54WNK 71452454 IC50 = 10.2 nM T67684 CPO41L 71452455 IC50 = 50.2 nM T67684 CYF3R2 71452456 IC50 = 158.9 nM T67684 C5WK8L 71452756 Ki = 0.13 nM T67684 CK81FI 71452793 Ki = 20.1 nM T67684 CG4ZX5 71454212 IC50 < 5 nM T67684 CSJ16R 71454213 IC50 < 5 nM T67684 CRMC04 71454214 IC50 < 5 nM T67684 CZS9G3 71454215 IC50 = 51.9 nM T67684 CR41KC 71454216 IC50 < 5 nM T67684 C5OBD0 71454217 IC50 = 579.3 nM T67684 CX26PA 71454562 Ki = 58.8 nM T67684 CX35MW 71454563 Ki = 0.38 nM T67684 C6G2HC 71455894 Ki = 1728 nM T67684 CQ98SO 71455965 IC50 = 27.5 nM T67684 CWZ6X0 71455966 IC50 < 5 nM T67684 C9N0HT 71455967 IC50 < 5 nM T67684 CS4TY5 71455968 IC50 = 45.3 nM T67684 CLWS62 71455969 IC50 = 142.6 nM T67684 CVI7S2 71457690 Ki = 2268 nM T67684 CP7JI0 71457691 Ki = 360 nM T67684 C3Z9KW 71457770 IC50 = 68.9 nM T67684 C63TRO 71457771 IC50 = 70.4 nM T67684 C56DYG 71457818 IC50 > 3300 nM T67684 CK5T4P 71459604 Ki = 1727 nM T67684 CQ64EL 71459689 IC50 = 197.3 nM T67684 CNKD53 71459690 IC50 < 5 nM T67684 C8Q2FH 71459691 IC50 = 82.2 nM T67684 CH9R6O 71459724 IC50 = 13.3 nM T67684 C8NWX4 71459909 Ki = 630.96 nM T67684 C2OIW1 71461631 IC50 = 315.4 nM T67684 CG8F1C 71461681 Ki = 27.8 nM T67684 C1Y9IC 71463063 Ki = 1225 nM T67684 CKG3U2 71463133 IC50 > 3300 nM T67684 CCR43M 71463134 IC50 = 392.4 nM T67684 C27RGM 71463135 IC50 = 44.9 nM T67684 C3AKB0 71463136 IC50 = 33.4 nM T67684 C8U1RC 71558565 IC50 = 1.585 nM T67684 C68UAI 71574174 Ki > 100000 nM T67684 C3MJ7B 71575027 Ki = 4070 nM T67684 CN82HY 71575122 Ki = 31100 nM T67684 CY1Q9O 71575447 Ki = 2840 nM T67684 CNS4V8 71575552 Ki > 100000 nM T67684 CM9SQ2 71575553 Ki > 100000 nM T67684 C89MPL 71575652 Ki = 4890 nM T67684 CM8UN7 71598549 IC50 > 30000 nM T67684 C1OE9J 71607097 IC50 > 30000 nM T67684 C3FQY2 71806339 IC50 > 10000 nM T67684 C4O5DN 72543915 IC50 = 0.631 nM T67684 C2XN9T 72543916 IC50 = 0.1 nM T67684 C9Y8CK 72543917 IC50 = 3.162 nM T67684 C3JED9 72543918 IC50 = 6.31 nM T67684 CAOG07 72545051 IC50 = 2.512 nM T67684 CJ2KM9 72545052 IC50 = 39.81 nM T67684 CPX8Q9 72545053 IC50 = 39.81 nM T67684 CHE5O6 72545089 Ki > 100000 nM T67684 CI6D4E 72545091 Ki > 100000 nM T67684 CKFW54 72545094 Ki > 100000 nM T67684 CWLO54 72545096 Ki > 100000 nM T67684 C5D4PA 72545098 Ki > 100000 nM T67684 C5XAE1 72545280 IC50 = 3.162 nM T67684 CY19JK 72545281 IC50 = 0.07943 nM T67684 CPU47R 72545282 IC50 = 0.0631 nM T67684 C1OPD2 72545283 IC50 < 0.03981 nM T67684 COH3J2 72545284 IC50 = 3.162 nM T67684 C0IX9Q 72545285 IC50 = 0.1585 nM T67684 CR39AG 72545326 Ki > 100000 nM T67684 C5HLF7 72545329 Ki > 100000 nM T67684 C45AZH 72545525 IC50 = 0.1259 nM T67684 CC38QM 72545526 IC50 = 0.0631 nM T67684 CQ6DW8 72545527 IC50 < 0.03981 nM T67684 CO3Z6K 72545528 IC50 = 0.05012 nM T67684 CTF30A 72545529 IC50 < 0.03162 nM T67684 CZN09L 72545530 IC50 = 0.1585 nM T67684 C84MRZ 72545782 IC50 = 1 nM T67684 C1NJ7R 72545783 IC50 = 0.5012 nM T67684 C1DP7G 72545784 IC50 = 0.05012 nM T67684 C3YG9K 72545785 IC50 = 0.1995 nM T67684 CH9ZP8 72545786 IC50 = 0.2512 nM T67684 CI6XY8 72545787 IC50 = 0.1259 nM T67684 CQ7OC5 72546023 IC50 = 100 nM T67684 C8FA0M 72546024 IC50 < 0.0631 nM T67684 CV5J7N 72546025 IC50 = 0.1585 nM T67684 CFD1H4 72546026 IC50 = 0.1 nM T67684 C4A3PY 72546028 IC50 = 0.3981 nM T67684 CN8TW2 72546260 IC50 = 12.59 nM T67684 CC52HE 72546261 IC50 = 0.1 nM T67684 CK4F2N 72546262 IC50 = 0.1585 nM T67684 CP94NR 72546263 IC50 = 0.2512 nM T67684 C89PYX 72546264 IC50 = 0.3981 nM T67684 C71AHG 72546492 IC50 = 25.12 nM T67684 COP12E 72546493 IC50 = 0.07943 nM T67684 CJ4C2D 72546494 IC50 = 0.3162 nM T67684 CREN32 72546495 IC50 = 10 nM T67684 CAEH63 72546496 IC50 = 0.1585 nM T67684 CWZ5C1 72546735 IC50 = 31.62 nM T67684 CNI4M9 72546736 IC50 = 0.1995 nM T67684 CY9NF4 72546737 IC50 = 2.512 nM T67684 CO95EP 72546738 IC50 = 0.631 nM T67684 CGSC63 72546739 IC50 = 0.1585 nM T67684 C59UXR 72546991 IC50 = 0.1585 nM T67684 CT0UB8 72546992 IC50 < 0.1259 nM T67684 CPQG94 72546993 IC50 = 0.2512 nM T67684 CKYM94 72546994 IC50 = 0.5012 nM T67684 CBM9V6 72546995 IC50 = 0.631 nM T67684 CND3O9 72547252 IC50 = 0.7943 nM T67684 C8V2TP 72547253 IC50 = 2.512 nM T67684 CCG30V 72547254 IC50 = 0.2512 nM T67684 C41FJI 72547255 IC50 = 0.7943 nM T67684 C7DL1J 72547256 IC50 = 0.3981 nM T67684 CXE9Y3 72547497 IC50 = 1 nM T67684 C4U8VC 72547498 IC50 = 0.7943 nM T67684 CBE0A1 72547499 IC50 = 2.512 nM T67684 C9R4GU 72547500 IC50 = 0.1995 nM T67684 C4YU3W 72547501 IC50 = 0.7943 nM T67684 CWH6T3 72548703 IC50 = 0.73 nM T67684 CG6Q8S 72712267 Ki = 0.3162 nM T67684 C27VLK 72712269 Ki = 0.0631 nM T67684 C7GS9W 72712271 Ki = 0.05012 nM T67684 C7FUP3 72712275 Ki = 1.585 nM T67684 C6F9EJ 72712473 Ki = 5.012 nM T67684 CT68WC 72712475 Ki = 1.995 nM T67684 CC65OA 73213195 Ki > 10000 nM T67684 CW83DK 73213196 Ki > 10000 nM T67684 C46HUP 73345823 Ki = 5.97 nM T67684 CRG9J8 73346332 Ki = 1782 nM T67684 CK0HR9 73346334 Ki = 2155 nM T67684 C6J0TM 73346336 Ki = 1301 nM T67684 CY60RD 73347826 Ki = 2119 nM T67684 C58SJG 73349591 Ki > 100000 nM T67684 CA6Z1P 73349592 Ki > 100000 nM T67684 C9Z1FO 73350398 Ki = 109 nM T67684 CDS4F1 73350931 Ki = 1058 nM T67684 CA8L9Y 73351145 Ki > 100000 nM T67684 CFM9Z0 73353378 Ki = 11.2 nM T67684 C4F7VK 73355415 Ki = 466 nM T67684 CX7ZV3 73356454 Ki = 0.543 nM T67684 CHV3W1 73774630 EC50 > 30000 nM T67684 C2E7QW 75201901 Ki > 10000 nM T67684 C8IDL3 75306277 Ki > 1000 nM T67684 CC4NP6 75356563 Ki = 4100 nM T67684 C1F0IU 76309737 IC50 = 318 nM T67684 C2NE1Q 76309753 IC50 = 154.4 nM T67684 CU5D8H 76309755 IC50 = 720.7 nM T67684 C42UQX 76309756 IC50 = 1161.3 nM T67684 CO2N6P 76309757 IC50 = 57.3 nM T67684 CUB3I6 76309856 IC50 = 7.943 nM T67684 C43NME 76313419 IC50 > 10000 nM T67684 CZ80LO 76313453 IC50 = 407.2 nM T67684 CFP71X 76313455 IC50 = 971.7 nM T67684 CNI0G8 76313457 IC50 = 776.3 nM T67684 CQ2AF0 76316968 IC50 = 137.4 nM T67684 CD3GN5 76316970 IC50 = 74.5 nM T67684 CP7T1M 76320689 IC50 = 342.1 nM T67684 CZ6C0O 76320691 IC50 = 713.9 nM T67684 CL7U5W 76320693 IC50 = 1143.6 nM T67684 CHZ0P7 76320694 IC50 = 261.6 nM T67684 CFR0L7 76324303 IC50 = 134 nM T67684 C6JZ5B 76324304 IC50 = 19 nM T67684 C94FIP 76324333 IC50 = 42.3 nM T67684 CN2S3T 76324335 IC50 = 2310.7 nM T67684 CA42PY 76324336 IC50 = 108 nM T67684 CB3M1C 76327869 IC50 < 10 nM T67684 C7GJ0Z 76327870 IC50 = 135 nM T67684 C9ATZ7 76327899 IC50 = 56.6 nM T67684 CQ94CR 76327901 IC50 = 2135.4 nM T67684 CUQ4W3 76327902 IC50 = 428.3 nM T67684 CJFI50 76327903 IC50 = 136.9 nM T67684 CGD90N 76331522 IC50 > 10000 nM T67684 CB46FR 76331543 IC50 = 109 nM T67684 CRH70L 87142783 Ki = 0.631 nM T67684 C2BM9L 89768534 EC50 > 30000 nM T67684 CB4Y7R 89768546 EC50 > 30000 nM T67684 CYX9R8 89777050 EC50 > 10000 nM T67684 C5MR9K 89777151 EC50 > 30000 nM T67684 C5UF4C 90666101 Ki = 0.39 nM T67684 CDI39M 90666102 Ki = 2.2 nM T67684 CU2FI1 90666103 Ki = 3.7 nM T67684 C18GXP 90666104 Ki = 18 nM T67684 C87KZI 90666105 Ki = 26 nM T67684 CBR34H 90666106 Ki = 10 nM T67684 CWG37L 90666107 Ki > 73 nM T67684 C30FIA 90666108 Ki = 22 nM T67684 CV61GN 90666109 Ki = 76 nM T67684 C0SIZ8 90666110 Ki = 8.3 nM T67684 C0FH6V 90666111 Ki = 4.8 nM T67684 CZ8I0G 90666112 Ki = 2 nM T67684 C6LB4R 90666113 Ki = 38 nM T67684 C5MCU0 90666114 Ki = 4.4 nM T67684 C0ZCW5 90666115 Ki = 1.1 nM T67684 CC5I0L 90666116 Ki = 2 nM T67684 CIZ46C 90666117 Ki = 4.4 nM T67684 C7WR2F 90666118 Ki = 9.2 nM T67684 C6KU1V 90666119 Ki = 4.3 nM T67684 CK68NB 90666120 Ki = 1.3 nM T67684 CEV61D 90666121 Ki = 8.9 nM T67684 CZ4P0B 90666122 Ki = 36 nM T67684 CV52KY 90666123 Ki = 3.1 nM T67684 C4RUP2 101882890 Ki = 1.096 nM T67684 CC3YS5 118706050 Ki > 100000 nM T67684 C6DXV9 118706052 Ki > 100000 nM T67684 CL4EO9 118706054 Ki = 26915.35 nM T67684 C4JY5S 118719502 IC50 > 30000 nM T67684 CI8CR0 118719920 Ki = 93.33 nM T67684 CV1WX5 118719921 Ki = 4.677 nM T67684 CIAG59 118719922 Ki = 0.7943 nM T67684 CC5Q8Y 118719923 Ki = 10 nM T67684 CC8R6U 118719924 Ki = 44.67 nM T67684 CT8KO4 118719925 Ki = 11748.98 nM T67684 C16DHZ 118719926 Ki = 1905.46 nM T67684 CLA06I 118719927 Ki = 630.96 nM T67684 CF20SR 118719928 Ki = 199.53 nM T67684 C6N7HV 118719929 Ki = 575.44 nM T67684 C64BIA 118719930 Ki = 338.84 nM T67684 CG4ZV5 118719931 Ki = 57.54 nM T67684 C05OBV 118723724 Ki > 100000 nM T67684 C37MUF 118728610 IC50 = 15 nM T67684 C96QNO 118728611 IC50 = 738.6 nM T67684 CTY76J 118737348 Ki = 0.1585 nM T67684 C6IMH9 118737349 Ki = 0.631 nM T67684 CPG45H 118737350 Ki = 1.259 nM T67684 CUE90B 118737351 Ki = 0.5012 nM T67684 C1DZ2G 118737352 Ki = 0.3162 nM T67684 C5VXT3 118737353 Ki = 6.31 nM T67684 CP37MC 118737354 Ki = 3.162 nM T67684 CGZX73 118737355 Ki = 0.7943 nM T67684 CB8J7S 118737356 Ki = 0.3162 nM T67684 CF1HQ8 118737357 Ki = 0.1995 nM T67684 CRE4M1 118737358 Ki = 1 nM T67684 CUN9G8 118737359 Ki = 7.943 nM T67684 CP6WF1 118737360 Ki = 1.995 nM T67684 COS3K9 121304408 Ki = 426.58 nM T67684 C4RD9Y 121304424 Ki = 549.54 nM T67684 C1PKR0 121304441 Ki = 380.19 nM T67684 CC3MP6 121304452 Ki = 302 nM T67684 CW68KD 121304458 Ki = 2041.74 nM T67684 CVA9F4 121304464 Ki = 275.42 nM T67684 COB2X5 121304477 Ki = 1230.27 nM T67684 CW51NQ 121304485 Ki = 275.42 nM T67684 C7NLV2 121304500 Ki = 891.25 nM T67684 CQ2UM4 121304538 Ki = 190.55 nM T67684 CN05ZQ 121304574 Ki = 354.81 nM T67684 CU0M7B 121304590 Ki = 1148.15 nM T67684 CX5MO3 121304598 Ki = 229.09 nM T67684 C12GJP 121304609 Ki = 1479.11 nM T67684 C31AEQ 121304649 Ki = 426.58 nM T67684 C2VTK5 121304654 Ki = 186.21 nM T67684 C5HQ4S 121304867 Ki = 2089.3 nM T67684 C1FB4S 122194235 Ki = 0.73 nM T67684 CH24YZ 122194236 Ki = 0.34 nM T67684 C8GP3F 122194237 Ki = 1.1 nM T67684 CX90IL 122194369 Ki = 5260 nM T67684 CU0B9P 122194370 Ki = 640 nM T67684 C79UOH 122194371 Ki > 10000 nM T67684 CMY91C 122194372 Ki = 3290 nM T67684 CCDI50 122194373 Ki = 4600 nM T67684 C3JI4Q 122194374 Ki = 370 nM T67684 CA6M5R 122194375 Ki > 30000 nM T67684 C7M1QH 122194376 Ki = 1540 nM T67684 C1JB0D 122194377 Ki = 4030 nM T67684 CD5NB9 122194378 Ki = 2300 nM T67684 C8O1QD 122194379 Ki > 10000 nM T67684 CFYZ56 122194380 Ki = 3550 nM T67684 COP38R 122195446 IC50 = 4170 nM T67684 CJM64P 122195453 IC50 = 4168.69 nM T67684 CB91PC 122195454 IC50 = 58000 nM T67684 CIV7R0 126533969 Ki = 1445.44 nM T67684 CIAD86 126534204 Ki = 1096.48 nM T67684 C4R7XU 126534291 Ki = 2187.76 nM T67684 CVBX50 126534373 Ki = 245.47 nM T67684 C0WUJ5 126534771 Ki = 1258.93 nM T67684 C9Q0VB 126535075 Ki = 478.63 nM T67684 CZ61LK 127034966 EC50 > 5011.87 nM T67684 CA0SN5 127034967 EC50 > 5011.87 nM T67684 CU9C4S 127041952 Ki = 1000 nM T67684 CJ2O5A 127044078 EC50 > 10000 nM T67684 CJ94GK 129316454 EC50 > 10000 nM T67684 C50GOC 130442480 Ki = 9200 nM T67684 CM04RF 130442572 Ki > 10000 nM T67684 CFXL21 132060812 Ki = 2369 nM T67684 CAVB41 132584404 Ki > 10000 nM T67684 CR8HL3 134134147 Ki = 676.08 nM T67684 CBU81N 134149168 Ki = 661 nM T67684 C0S2VH 134150637 Ki = 676.08 nM T67684 C6NYU2 134150754 Ki = 630.96 nM T67684 C1GY2T 135156251 EC50 > 10000 nM T67684 C4UX2M 135430667 Ki = 3090.3 nM T67684 CGS61F 137553161 Ki = 3000 nM T67684 CI5SL0 137633162 Ki = 140 nM T67684 CD91UT 137634680 Ki = 14000 nM T67684 COI42G 137635637 EC50 = 3700 nM T67684 C6QB9W 137635734 Ki = 6606.93 nM T67684 CX8O0V 137636308 Ki = 7079.46 nM T67684 CRH92D 137636829 Ki = 8700 nM T67684 CWT0D8 137637047 Ki = 12000 nM T67684 C7VUW4 137637944 IC50 = 380 nM T67684 CY8Q1V 137638270 IC50 = 782 nM T67684 CFDB34 137639384 Ki = 5800 nM T67684 C4YJ1T 137639541 Ki = 42000 nM T67684 CVIA23 137640095 Ki = 4700 nM T67684 CZ4TA9 137640201 Ki = 3019.95 nM T67684 CX4A3N 137640511 Ki = 14125.38 nM T67684 C2POD8 137640878 Ki = 43000 nM T67684 CYW61U 137641749 IC50 > 16000 nM T67684 C8ZDW1 137642318 Ki = 11000 nM T67684 C4Q6ZM 137642607 Ki = 4677.35 nM T67684 CW4IJ1 137644950 Ki = 75000 nM T67684 C0KL6Q 137644962 Ki = 6760.83 nM T67684 CPCY48 137645406 Ki = 514 nM T67684 CG8P6I 137645938 Ki = 1348.96 nM T67684 CO58KT 137646451 Ki = 620 nM T67684 CJIU91 137647528 Ki = 12000 nM T67684 C2XMK6 137647734 IC50 = 365 nM T67684 CB9PL0 137648038 Ki = 2000 nM T67684 C3LC9W 137648483 Ki = 4000 nM T67684 CBN1K6 137650836 Ki = 199.53 nM T67684 C6WS1K 137653145 Ki = 25000 nM T67684 CFZS94 137653227 Ki = 20000 nM T67684 CWF8R1 137653324 Ki = 5800 nM T67684 C8XJO5 137653498 Ki = 690 nM T67684 C61WAG 137654353 IC50 = 660 nM T67684 CC7GE8 137654674 Ki = 13000 nM T67684 CWOV78 137655063 IC50 = 404 nM T67684 CUC54G 137655636 Ki = 501.19 nM T67684 CUKT36 137655796 EC50 = 10000 nM T67684 CRY40J 137655938 IC50 = 610 nM T67684 CUZ2V9 137656894 Ki = 3900 nM T67684 CQ2H0S 137657830 Ki = 210 nM T67684 CWSA41 137658091 Ki = 16000 nM T67684 C6E0JP 137659594 Ki = 41 nM T67684 C4BAP3 137660708 Ki = 21000 nM T67684 C7NJH0 137661079 Ki = 24000 nM T67684 C68QKL 137661317 Ki = 15.49 nM T67684 CDA8V2 137661377 Ki = 2344.23 nM T67684 C41ZYJ 137701968 EC50 > 30000 nM T67684 C9J1ZO 142416754 IC50 = 11000 nM T67684 C58KQF 142416884 IC50 > 33000 nM T67684 C68OXK 142416914 IC50 > 17000 nM T67684 CO7DK2 142416967 IC50 > 33000 nM T67684 COG04E 145950432 IC50 = 9600 nM T67684 C3OMF2 145951963 IC50 = 8800 nM T67684 CPW52X 145954567 IC50 = 23000 nM T67684 C0HN4S 145955917 IC50 = 10000 nM T67684 C4G6XJ 145956824 IC50 = 13000 nM T67684 CXHM49 145958111 IC50 = 32 nM T67684 CBC1T9 145958296 IC50 = 1100 nM T67684 CH47WN 145959135 IC50 > 16000 nM T67684 CI8Q2V 145960175 IC50 = 770 nM T67684 C38OTS 145960427 Ki = 416.87 nM T67684 C06LVP 145960466 Ki = 19.95 nM T67684 CSV5D4 145960592 Ki = 269.15 nM T67684 C4KH9G 145960827 Ki = 104.71 nM T67684 CJI6G2 145961125 Ki = 2630.27 nM T67684 CK7OJ5 145961126 Ki = 1621.81 nM T67684 C0XL7S 145961152 Ki = 14454.4 nM T67684 C3WFT9 145961161 Ki = 43.65 nM T67684 CJ50OV 145961495 Ki = 398.11 nM T67684 CAH97Y 145961981 Ki = 1548.82 nM T67684 CH1AE6 145962050 Ki = 1698.24 nM T67684 CG16NQ 145963288 Ki = 616.6 nM T67684 C1DW4U 145983928 IC50 > 100000 nM T67684 CMJ46R 145990794 IC50 > 100000 nM T67684 C9PS8N 145993117 IC50 > 100000 nM T67684 C0Z6YX 145993493 IC50 > 100000 nM T67684 CC2G1V 146025727 Ki = 2700 nM T67684 C6P3SR 153287553 Ki > 10000 nM T67684 CV9G7Z 153287572 Ki > 10000 nM T67684 CO85KL 153287574 Ki > 10000 nM T67684 CJKG35 155510347 Ki = 4360 nM T67684 C8IXK6 155511112 Ki = 390 nM T67684 CY83UA 155511167 Ki = 60 nM T67684 CSR04X 155512177 Ki = 1.1 nM T67684 CCB34Y 155512243 Ki = 17 nM T67684 C2BDK6 155513985 Ki = 954.99 nM T67684 CK30XC 155514683 Ki = 19 nM T67684 C6JSC8 155515662 Ki = 90 nM T67684 C4OGI7 155515788 Ki = 2.8 nM T67684 CUM2N4 155515982 Ki = 25000 nM T67684 CJG12Y 155516095 Ki = 1150 nM T67684 C53FKW 155516382 Ki = 660.69 nM T67684 CI24NW 155516845 Ki = 550 nM T67684 C0JM8H 155518181 Ki = 70 nM T67684 C0MT4Q 155519740 Ki = 38.02 nM T67684 CUSA24 155519891 Ki > 10000 nM T67684 C4B7VK 155520267 Ki = 350 nM T67684 C1R9WB 155520414 Ki = 0.44 nM T67684 C3R6GZ 155520947 Ki = 1.7 nM T67684 CPVA65 155521382 Ki = 1479.11 nM T67684 C9N3JA 155521639 Ki = 1560 nM T67684 C7HPL3 155521847 Ki = 260 nM T67684 CFVP27 155521893 Ki = 16.22 nM T67684 CL9ET5 155522354 Ki = 6760.83 nM T67684 CI2RK6 155523171 Ki = 6.5 nM T67684 CL6O1R 155523647 Ki = 13.49 nM T67684 C38PTA 155523888 Ki = 2691.53 nM T67684 C8AMH9 155524478 Ki = 250 nM T67684 C6PFY7 155524809 Ki = 290 nM T67684 C5P1YE 155525064 Ki = 1380.38 nM T67684 CDQ89Y 155525097 Ki = 13.18 nM T67684 CBK1S6 155525654 Ki = 0.65 nM T67684 C7EIK1 155525691 Ki = 570 nM T67684 CBK0Y7 155528269 Ki = 5495.41 nM T67684 CPG08Y 155528419 Ki = 420 nM T67684 CRPY78 155529196 Ki = 20 nM T67684 CIA9P5 155530272 Ki = 1.9 nM T67684 C6K5WZ 155531077 IC50 = 1.585 nM T67684 C1U3VP 155535038 Ki = 20 nM T67684 C7CU8J 155535606 Ki = 28.18 nM T67684 CK91NV 155535972 Ki = 140 nM T67684 CB79ZW 155536080 Ki > 10000 nM T67684 C2XN8P 155536739 Ki = 50 nM T67684 C9ZW3N 155537081 Ki = 4.7 nM T67684 CR17JS 155539026 Ki = 184 nM T67684 CV2NG9 155539712 Ki = 28.18 nM T67684 CG3A9Y 155539770 Ki = 0.4 nM T67684 CMUF93 155540312 Ki = 2.3 nM T67684 CY2L3J 155540315 Ki = 1280 nM T67684 CK70MJ 155541812 Ki = 2.6 nM T67684 C7DMY9 155542295 Ki = 0.51 nM T67684 CL7ZA6 155542839 Ki = 1.5 nM T67684 CS5YB1 155543344 Ki = 5011.87 nM T67684 COV93Z 155543943 Ki = 151.36 nM T67684 CI8KA5 155544834 Ki = 42 nM T67684 C2CB8H 155548585 Ki = 1258.93 nM T67684 CMS50Z 155549803 Ki = 0.86 nM T67684 C1XIA4 155549890 Ki = 1320 nM T67684 C1UA2M 155550149 Ki = 2.6 nM T67684 C9KBH7 155550435 Ki = 27.54 nM T67684 CRIJ70 155550631 Ki = 48.98 nM T67684 CR8XF7 155551306 Ki = 130 nM T67684 C6RK4Q 155551382 Ki = 3.8 nM T67684 CW92JZ 155551421 Ki = 2800 nM T67684 COF49W 155551902 Ki = 5370.32 nM T67684 CX8JA1 155552185 Ki = 37000 nM T67684 CXZQ46 155552922 Ki = 10000 nM T67684 CE70NU 155553089 Ki = 270 nM T67684 CN4ZH3 155553222 Ki = 7.8 nM T67684 CS1DK6 155554149 Ki = 19 nM T67684 C7TF1D 155554261 Ki = 1584.89 nM T67684 C73DFN 155554567 Ki = 154.88 nM T67684 C1TDY8 155556289 Ki = 44.67 nM T67684 C2D3SP 155557118 Ki = 1148.15 nM T67684 C75PXS 155559290 Ki > 10000 nM T67684 CEAD84 155559740 Ki = 1621.81 nM T67684 CP2U8A 155560012 Ki = 645.65 nM T67684 CU3TF1 155560139 Ki = 776.25 nM T67684 CCO15D 155560304 Ki = 61.66 nM T67684 CMX98Q 155562285 Ki = 8 nM T67684 C7P2OG 155562295 Ki = 1020 nM T67684 CDYV69 155562882 Ki = 300 nM T67684 C8WE2F 155563061 Ki = 2760 nM T67684 C4N9GU 155563428 Ki = 5900 nM T67684 CSO40U 155564307 Ki = 41 nM T67684 C2G7UH 155565074 Ki = 220 nM T67684 CVLR58 155565285 Ki > 10000 nM T67684 C9AF7I 155565770 Ki = 60 nM T67684 CDS7K2 155566289 Ki = 109.65 nM T67684 CY30EN 155567379 Ki = 35.48 nM T67684 C38QRW 155568227 Ki = 81 nM T67684 CKS4A0 155568815 Ki = 0.86 nM T67684 C3N9VU 10251906 Ki > 500 nM T67684 C12RSP 11364984 IC50 = 39.81 nM T67684 C9RLJ3 3661 Ki = 0.53 nM T67684 CD6OK3 44455198 Ki = 10.3 nM T67684 CZCS12 44573305 IC50 = 501.19 nM T67684 D01JXM 46222048 Ki > 1000 nM T67684 D01UDC 9815331 Ki = 680 nM T67684 D02BOW 5926 Ki = 2398.83 nM T67684 D02EXX 3013846 Ki = 130 nM T67684 D02KZD 71598521 IC50 > 30000 nM T67684 D02ZPV 10125445 Ki = 3.162 nM T67684 D03DKZ 42633508 EC50 > 30000 nM T67684 D04XNH 44318851 Ki = 11400 nM T67684 D05EML 21847 IC50 < 1 nM T67684 D05YBO 3013847 Ki = 1000 nM T67684 D05ZUX 44207909 Ki >= 1000 nM T67684 D06IUC 6508730 Ki = 24 nM T67684 D07GPQ 132947 Ki = 38.02 nM T67684 D07QGQ 135466875 Ki = 970 nM T67684 D09RPR 16737207 Ki > 10000 nM T67684 D09YBC 3013845 Ki = 1250 nM T67684 D0A2KT 3014059 Ki = 0.22 nM T67684 D0AR0H 6508724 Ki = 30 nM T67684 D0C9ZE 10105296 Ki = 1300 nM T67684 D0F5LH 4634 Ki = 0.78 nM T67684 D0FF6S 16038374 IC50 > 10000 nM T67684 D0G4CG 4629 EC50 = 1800 nM T67684 D0H8XV 12963076 Ki = 3388.44 nM T67684 D0HP1O 119357 Ki = 66.07 nM T67684 D0I2XG 135494454 Ki = 230 nM T67684 D0I9LU 2229 Ki = 851.14 nM T67684 D0IL1B 3494 IC50 = 0.2512 nM T67684 D0J4DJ 135423423 Ki = 1330 nM T67684 D0JV2S 3008304 EC50 = 6380 nM T67684 D0L1XR 4630 EC50 = 210 nM T67684 D0L5MW 181743 Ki > 10000 nM T67684 D0M5ZE 5311416 Ki = 1995.26 nM T67684 D0P1FJ 71128 Ki = 7.7 nM T67684 D0Q2VN 77157 Ki = 1.1 nM T67684 D0T2RY 9948320 Ki >= 1000 nM T67684 D0TX8W 594590 Ki > 19952.62 nM T67684 D0WO3A 4141 Ki = 6165.95 nM T67684 D0X7HD 11184481 Ki = 8300 nM T67684 D0Z5RQ 656392 IC50 = 126 nM T67684 D0Z6VT 71737672 EC50 = 2100 nM T88975 D0L0ZF 5663 IC50 = 10700 nM T88975 D0NJ3V 4680 Ki = 279 nM T88975 D0R4UW 449193 IC50 > 100000 nM T88975 D0Y9ZE 4197 IC50 = 3600 nM T88975 D0Z7ZM 135398744 IC50 = 26000 nM T88975 D01LCC 17754438 IC50 > 10000 nM T88975 D03QJL 3671 IC50 = 299000 nM T88975 D0A9IY 135564558 IC50 > 10000 nM T88975 D0WS3T 72706254 IC50 > 10000 nM T88975 C9LH4S 371187 IC50 = 3980 nM T88975 C1B6ZL 662965 IC50 > 50000 nM T88975 COS03W 1204288 IC50 = 10500 nM T88975 CK8DT9 1205767 IC50 = 9460 nM T88975 C3D0HY 1232680 IC50 = 80000 nM T88975 CPXC25 1368101 IC50 = 39810 nM T88975 C8JLO0 2243267 IC50 > 10000 nM T88975 CNMR07 3395707 IC50 = 27000 nM T88975 CK12OT 3814427 IC50 = 1110 nM T88975 CC3LA4 4672917 IC50 = 21300 nM T88975 C5P0LU 4672918 IC50 = 29300 nM T88975 CI7K0P 6918667 IC50 > 101000 nM T88975 CP1GO7 6918668 IC50 = 78100 nM T88975 C87WYR 6918795 IC50 = 42200 nM T88975 CRGE51 6918796 IC50 > 79900 nM T88975 CUP4M8 6918797 IC50 = 44500 nM T88975 C0LRO8 6918798 IC50 > 68000 nM T88975 C53ESK 6918799 IC50 > 73000 nM T88975 CU1E0G 6918800 IC50 > 101000 nM T88975 CI5GD6 9816296 IC50 = 96 nM T88975 C4J2XE 9836643 IC50 = 101000 nM T88975 C5YQB0 9859898 IC50 = 110000 nM T88975 C0Q5VN 9880010 IC50 > 101000 nM T88975 CWD1F6 9880288 IC50 > 101000 nM T88975 CC05QE 9901606 IC50 > 101000 nM T88975 CBA29H 9922545 IC50 = 94000 nM T88975 CKF4C2 9922691 IC50 > 101000 nM T88975 C70AMC 9924305 IC50 = 7470 nM T88975 CKI6N2 9924468 IC50 = 11800 nM T88975 C6AZ5F 9924709 IC50 > 101000 nM T88975 CX1UV7 9946954 IC50 = 8570 nM T88975 C7OP5A 9947052 IC50 = 5580 nM T88975 CJO0X4 9966737 IC50 = 6130 nM T88975 CFP1Y5 9966830 IC50 > 101000 nM T88975 C9NKY4 9967652 IC50 > 101000 nM T88975 CI6AX1 9968005 IC50 = 2650 nM T88975 C7PCS8 9968050 IC50 = 30680 nM T88975 CFB48Q 9968370 IC50 > 101000 nM T88975 CU73AJ 9968471 IC50 > 101000 nM T88975 C0AP8O 9969020 IC50 = 16980 nM T88975 C12LED 10109572 IC50 > 101000 nM T88975 C2PBD6 10131447 IC50 = 14800 nM T88975 C5HC2X 10182563 IC50 = 31600 nM T88975 C3GN8K 10200432 IC50 = 10800 nM T88975 C8JR4W 10221093 IC50 = 89000 nM T88975 CFGO46 10221904 IC50 = 12700 nM T88975 CQ61CV 10268304 IC50 = 45100 nM T88975 C1QU2B 10268305 IC50 = 11200 nM T88975 CH9C4K 10269859 IC50 = 20540 nM T88975 CR92JY 10270352 IC50 > 101000 nM T88975 C7CHR0 10270536 IC50 = 16700 nM T88975 C2AE6K 10340179 IC50 = 1.3 nM T88975 C3B1QP 11161553 IC50 = 3800 nM T88975 CU98NK 11518003 IC50 = 7.6 nM T88975 C9FB1N 11532490 IC50 = 150 nM T88975 CS2PA6 11545321 IC50 = 98 nM T88975 C3EM0P 11559345 IC50 = 8.5 nM T88975 C8R1NX 11566058 IC50 = 360 nM T88975 CO2GR1 11574595 IC50 = 53 nM T88975 C0P8DN 11596587 IC50 = 1.6 nM T88975 C3G1BO 11604203 IC50 = 27500 nM T88975 C69RXL 11655838 IC50 = 2.2 nM T88975 CR8CQ7 11669507 IC50 = 38500 nM T88975 C8YRP7 11955134 IC50 = 11300 nM T88975 CG3RA6 11955200 IC50 = 360 nM T88975 CL6F4C 11955614 Ki = 211 nM T88975 C1B4XD 11992634 IC50 > 2000 nM T88975 CPX16N 11993169 IC50 > 2000 nM T88975 CBX53H 12805021 IC50 = 2.9 nM T88975 CSX70H 15991588 Ki = 283 nM T88975 C08TUE 16102593 Ki < 100 nM T88975 C7GDQ8 16102594 Ki < 100 nM T88975 CJQA32 16102595 Ki > 100 nM T88975 CHAL10 16102596 Ki < 100 nM T88975 CX0EG2 16102597 Ki = 739 nM T88975 C6Z7GM 16102598 Ki = 161 nM T88975 C4JVF5 16102599 Ki = 271 nM T88975 CMR3A7 16102600 Ki = 141 nM T88975 CX1B4L 16102601 Ki = 162 nM T88975 CC0DP8 16102602 Ki = 77 nM T88975 CLH34A 16102603 Ki = 226 nM T88975 CK06QM 16102604 Ki = 48 nM T88975 C4TH8R 16102605 Ki = 273 nM T88975 C6X1VB 16102606 Ki = 152 nM T88975 C04SBT 16102607 Ki = 151 nM T88975 C9IK5Y 16102620 Ki < 100 nM T88975 CL6Y7J 16102621 Ki < 100 nM T88975 CNAW90 16102622 Ki = 214 nM T88975 C1GD3A 16102623 Ki = 720 nM T88975 CX43OI 16102624 Ki = 370 nM T88975 CA52VZ 16102625 Ki = 61 nM T88975 CH25WX 16102626 Ki = 121 nM T88975 C5V1LM 16102627 Ki = 302 nM T88975 CC21RZ 16102628 Ki = 199 nM T88975 C5SN6Y 16102629 Ki = 104 nM T88975 C3S2KA 16102630 Ki = 209 nM T88975 CYN39I 16666580 IC50 = 9210 nM T88975 C0HI2G 16666581 IC50 = 9010 nM T88975 CAW98T 16666618 IC50 = 75550 nM T88975 CD1VU8 16666619 IC50 = 1590 nM T88975 CJP10M 16666620 IC50 = 2500 nM T88975 CM91TF 16666621 IC50 = 6170 nM T88975 C4U3WX 16666622 IC50 = 4130 nM T88975 CXFT59 17757146 IC50 = 1700 nM T88975 CW96CH 21158737 IC50 = 0.33 nM T88975 C7RK1W 21920272 IC50 = 9830 nM T88975 CH7N9S 21920275 IC50 = 1710 nM T88975 CV04DH 21920370 IC50 = 47210 nM T88975 CW96SI 23624262 IC50 = 1260 nM T88975 CM3E7V 23647030 IC50 = 15 nM T88975 C0MO2Z 23647031 IC50 = 24 nM T88975 C46WZJ 23647032 IC50 = 44 nM T88975 CEJY54 23647042 IC50 = 22 nM T88975 C2CO7U 23647044 IC50 = 3.7 nM T88975 C3A7BX 23647045 IC50 = 101 nM T88975 C2YSQ6 23647046 IC50 = 1.2 nM T88975 C4M9BC 23647047 IC50 = 46 nM T88975 C7P2CZ 23647048 IC50 = 1.6 nM T88975 C09BFZ 23647049 IC50 = 38 nM T88975 CD56GP 23647050 IC50 = 130 nM T88975 C76IBZ 23647051 IC50 = 20 nM T88975 CE5PL6 23647052 IC50 = 69 nM T88975 C0IM7N 23647053 IC50 = 7.2 nM T88975 CE9L7Y 23647054 IC50 = 16 nM T88975 C8QZ0R 23647055 IC50 = 43 nM T88975 CED1K2 23647056 IC50 = 63 nM T88975 CN40CL 23647057 IC50 = 550 nM T88975 CBF94I 23647058 IC50 = 77 nM T88975 CBXC05 24424330 IC50 = 490 nM T88975 CAJ57O 24751843 IC50 = 72000 nM T88975 CL79TD 24751991 IC50 > 400000 nM T88975 C7QEC1 24772445 IC50 > 100000 nM T88975 CHX26Y 24772447 IC50 > 100000 nM T88975 C2LS4C 24772511 IC50 > 100000 nM T88975 CDU9R1 24772513 IC50 > 100000 nM T88975 CZF02U 24798187 IC50 = 67100 nM T88975 C2ET7F 24799903 IC50 = 6650 nM T88975 C0GHB4 24799905 IC50 = 140 nM T88975 CY9H4A 24799906 IC50 = 540 nM T88975 C3TJ2G 24799907 IC50 = 14120 nM T88975 C7ZH3R 24800081 IC50 = 5360 nM T88975 CM9DG6 24800082 IC50 = 1100 nM T88975 C9WGI4 24802717 IC50 = 3700 nM T88975 C0UY9O 24802801 IC50 = 22200 nM T88975 C73ABX 24802803 IC50 = 5740 nM T88975 C0LEU9 24802804 IC50 = 150 nM T88975 CA74HQ 24804333 IC50 = 140 nM T88975 CJGZ93 24804334 IC50 = 270 nM T88975 C20JRY 24804335 IC50 = 72 nM T88975 CG64YI 24804336 IC50 = 1.2 nM T88975 C39PBK 24804498 IC50 = 5.1 nM T88975 C20VHK 24871823 IC50 = 3530 nM T88975 C6EQG2 24963293 IC50 > 2000 nM T88975 C9TS3H 25018106 IC50 = 2850 nM T88975 CPIO29 25018348 IC50 = 10200 nM T88975 C2B4NM 25026184 IC50 = 1.7 nM T88975 C8YBW4 25055989 IC50 = 2370 nM T88975 CC58QZ 25055991 IC50 = 10840 nM T88975 CBL3C7 25056255 IC50 = 2000 nM T88975 CB79EW 25056256 IC50 = 3280 nM T88975 C7V4AS 25142306 IC50 = 5 nM T88975 C1MCK3 25142307 IC50 = 63 nM T88975 C4J0YD 25196719 IC50 = 3070 nM T88975 CICF39 42629702 IC50 = 2680 nM T88975 CM3X9S 42629827 IC50 > 1000 nM T88975 CQN26J 42629945 IC50 > 10000 nM T88975 C6O5FX 42630062 IC50 > 5000 nM T88975 C71ZNR 42630180 IC50 = 6900 nM T88975 C4RHY0 42630191 IC50 > 10000 nM T88975 CT6RS9 42630192 IC50 > 10000 nM T88975 CYZL43 42630317 IC50 > 10000 nM T88975 CH42OZ 42630318 IC50 > 10000 nM T88975 C7X5AH 42630437 IC50 > 10000 nM T88975 CQU19I 44180409 IC50 = 101000 nM T88975 CW8OB3 44243146 Ki > 10000 nM T88975 CMFN38 44351947 IC50 = 0.94 nM T88975 C7V8YH 44351948 IC50 = 2.8 nM T88975 CXC52L 44352035 IC50 = 2.3 nM T88975 C2V4KH 44352046 IC50 = 0.11 nM T88975 CKJ01T 44352047 IC50 = 3.1 nM T88975 CIM5Z7 44352055 IC50 = 0.11 nM T88975 CK7O1X 44352067 IC50 = 24 nM T88975 C6PZ2V 44352121 IC50 = 0.83 nM T88975 C6OJ4R 44352133 IC50 = 0.39 nM T88975 C13HPW 44393651 IC50 > 92000 nM T88975 CJ6GB5 44393709 IC50 = 280 nM T88975 CQP01D 44393950 IC50 = 49420 nM T88975 CU1CQ8 44394047 IC50 = 78000 nM T88975 C98UBL 44452447 Ki = 739 nM T88975 CPOZ04 44452603 Ki = 370 nM T88975 CVY0F4 44453752 IC50 = 24990 nM T88975 CGK59A 44453754 IC50 = 28500 nM T88975 CF73GI 44453781 IC50 = 10830 nM T88975 C7VW4N 44817564 IC50 = 13300 nM T88975 C36XLQ 46209046 IC50 > 30000 nM T88975 C2Q4YT 46209162 IC50 > 30000 nM T88975 CJOE41 46209386 IC50 > 30000 nM T88975 C5QCW8 46229955 IC50 = 1760 nM T88975 CFJ6O8 46229956 IC50 = 1440 nM T88975 CX85PB 46229957 IC50 = 1650 nM T88975 CG57XW 46229958 IC50 = 1260 nM T88975 CDFM64 46229998 IC50 = 840 nM T88975 CQEK64 46229999 IC50 = 1350 nM T88975 C4D5KO 46230000 IC50 = 660 nM T88975 CX56CQ 46230001 IC50 = 430 nM T88975 CCV17X 46230002 IC50 = 1340 nM T88975 COS0L1 46230055 IC50 = 640 nM T88975 CR0Y7J 46230056 IC50 = 2840 nM T88975 C5IMB2 46239424 Ki > 10000 nM T88975 CKR9P7 46239425 Ki > 10000 nM T88975 C3P2IN 46933992 IC50 >= 29000 nM T88975 CHA5Z0 49821469 IC50 > 1000 nM T88975 C1AYP0 49821627 IC50 > 500 nM T88975 C85AXR 49821714 IC50 > 1000 nM T88975 C0B8JE 49843464 Ki = 177 nM T88975 CMN05G 50901953 Ki = 1738 nM T88975 CZS03D 50902030 Ki = 449 nM T88975 CPL5E6 50902114 Ki = 136 nM T88975 CAD40F 50902119 Ki = 954 nM T88975 CD98UC 50902202 Ki = 1279 nM T88975 CXB85R 50902203 Ki = 1472 nM T88975 C9QLF2 50902206 Ki = 277 nM T88975 CH2Z1E 50902289 Ki = 968 nM T88975 C4HJL2 50902291 Ki = 727 nM T88975 C7EQ9Y 50902548 Ki = 99 nM T88975 C6A1IU 50902549 Ki = 149 nM T88975 CVM28N 50902550 Ki = 24 nM T88975 CN1P7Q 50902632 Ki = 828 nM T88975 C3Y2AV 50903255 Ki = 555 nM T88975 C6R4YN 50993785 IC50 = 10000 nM T88975 C0M6XL 50993786 IC50 = 10000 nM T88975 C0OR7K 53248667 IC50 = 2750 nM T88975 C24HYO 53248668 IC50 = 39600 nM T88975 CS3R1I 53248669 IC50 = 33500 nM T88975 C30RNE 53248670 IC50 = 41500 nM T88975 CS0ZD1 53324378 IC50 = 14.8 nM T88975 CHLA42 54576311 IC50 = 1290 nM T88975 C6DEG8 54576313 IC50 = 1190 nM T88975 CJF0K2 54576315 IC50 = 1940 nM T88975 CNW81G 54576317 IC50 = 1740 nM T88975 C9WEO5 54576525 IC50 = 2200 nM T88975 C1RJ7M 54580520 IC50 > 400000 nM T88975 CCXF36 54580521 IC50 = 7000 nM T88975 CZG36N 54580522 IC50 = 26000 nM T88975 C0NPM8 54580523 IC50 = 260000 nM T88975 C25VSX 54580524 IC50 > 400000 nM T88975 C0MN3D 54582527 IC50 = 3200 nM T88975 C6T1QX 54582528 IC50 = 210000 nM T88975 CW1X3G 54583497 IC50 > 400000 nM T88975 CN96IQ 54585432 IC50 > 400000 nM T88975 CH25CO 54586393 IC50 > 400000 nM T88975 C82LED 54586394 IC50 = 8900 nM T88975 CQ1H3C 54587403 IC50 = 15000 nM T88975 C28GAC 54587404 IC50 = 69000 nM T88975 CGF65A 54670110 IC50 > 30000 nM T88975 C90ZLC 54670399 IC50 = 208 nM T88975 C4TGL7 56648496 IC50 > 1000 nM T88975 CH6C3L 56648679 IC50 > 10000 nM T88975 CCY79V 56648680 IC50 = 5280 nM T88975 CNE96P 56648857 IC50 > 5000 nM T88975 CX86AQ 56648859 IC50 > 5000 nM T88975 CPC3T4 56654131 IC50 > 10000 nM T88975 C0YD3P 56928304 IC50 > 5000 nM T88975 C8RO6A 56929788 IC50 > 1000 nM T88975 C3ZRD5 56929886 IC50 = 6430 nM T88975 C2G9PX 57345604 IC50 = 970 nM T88975 CUS7R9 57385526 IC50 = 104200 nM T88975 CB17SC 57385767 IC50 = 54600 nM T88975 CH75PT 57385768 IC50 = 1800 nM T88975 C7EB5V 57386043 IC50 = 3400 nM T88975 CK81XA 57386556 IC50 = 3900 nM T88975 CD52CA 57391118 IC50 > 2000 nM T88975 CG3DF1 57392948 Ki > 10000 nM T88975 CE36TV 57394695 Ki > 10000 nM T88975 CB21SH 57398742 IC50 = 19800 nM T88975 C7VMN0 57398767 IC50 = 1450 nM T88975 C5BM4F 57400402 IC50 = 20700 nM T88975 CPA3D1 57403394 Ki > 10000 nM T88975 C4XMB6 58547809 IC50 > 30000 nM T88975 CEB3G9 58547814 IC50 > 30000 nM T88975 C08QVG 58547833 IC50 > 30000 nM T88975 CFVG67 58547863 IC50 > 30000 nM T88975 CYZA38 58548077 IC50 > 30000 nM T88975 CZI9U7 59227406 IC50 > 100000 nM T88975 C34SNK 59227413 IC50 > 100000 nM T88975 CVH8T2 59227421 IC50 > 100000 nM T88975 CWX3N7 59320301 IC50 = 1800 nM T88975 COC80E 59335994 IC50 = 6.9 nM T88975 CN62MK 59336034 IC50 = 10080 nM T88975 CB9GO8 59336035 IC50 = 40 nM T88975 C0EP5I 59341847 IC50 = 1250 nM T88975 CHQ28A 59341978 IC50 = 589 nM T88975 CJ0YB8 59351288 IC50 > 30000 nM T88975 CCA1H6 59351376 IC50 > 30000 nM T88975 CN57ZH 67426178 IC50 > 10000 nM T88975 CY8J3O 68181896 IC50 > 30000 nM T88975 C4ZEH9 68578314 IC50 = 78000 nM T88975 CUGH78 68654838 IC50 = 1584.89 nM T88975 COI2P3 70679302 IC50 > 30000 nM T88975 CU9GQ0 70681149 Ki = 540 nM T88975 CI9G8L 70683261 Ki = 224 nM T88975 C6BN5J 70685361 Ki > 100000 nM T88975 CK7Y2D 70686701 IC50 = 1630 nM T88975 CF6O3T 70687501 Ki = 148 nM T88975 CC43LF 71074083 IC50 > 10000 nM T88975 C4P0XT 71092344 IC50 = 6210 nM T88975 C6DAG4 71092519 IC50 > 30000 nM T88975 C9GR3L 71153436 IC50 = 7760 nM T88975 CR5NQ6 71450591 IC50 > 30000 nM T88975 CGD56M 71450592 IC50 > 30000 nM T88975 CZ1YN2 71452430 IC50 > 30000 nM T88975 CI1M8Q 71452431 IC50 > 30000 nM T88975 CX5D2O 71454197 IC50 > 30000 nM T88975 CJV1G2 71455939 IC50 > 30000 nM T88975 C8A4ME 71457746 IC50 > 30000 nM T88975 C3VKH8 71459650 IC50 > 30000 nM T88975 CT2D6E 71461384 IC50 > 30000 nM T88975 C13OKG 71517744 IC50 = 130 nM T88975 C54EWN 71517745 IC50 = 15 nM T88975 CKOZ85 71517907 IC50 = 11 nM T88975 CB0OK6 71517908 IC50 = 40000 nM T88975 CC8GZ6 71517909 IC50 = 360 nM T88975 CP9G6K 71517910 IC50 = 38000 nM T88975 CP6DN1 71517911 IC50 = 590 nM T88975 C6D7EY 71518079 IC50 = 1730 nM T88975 C83PUL 71518080 IC50 = 1520 nM T88975 CBJZ01 71518081 IC50 = 58 nM T88975 C7Q2GV 71518082 IC50 = 15 nM T88975 C40KMI 71518243 IC50 = 0.27 nM T88975 CJ36SE 71518244 IC50 = 2.7 nM T88975 C4GNJ3 71598545 IC50 > 1000 nM T88975 COWG10 71748255 IC50 = 14000 nM T88975 CZ0G2X 72165213 IC50 > 10000 nM T88975 C7XRY6 72190879 IC50 > 30000 nM T88975 C38UIK 72192868 IC50 = 71400 nM T88975 C5KPN6 72193179 IC50 > 100000 nM T88975 CBM61I 73293715 IC50 = 2870 nM T88975 CHR7D0 73334611 IC50 = 7470 nM T88975 C9ODB8 73387740 IC50 = 23600 nM T88975 C5X6GJ 73387742 IC50 > 20000 nM T88975 CT1E6V 73387743 IC50 = 8520 nM T88975 C7D1SJ 73387744 IC50 = 111900 nM T88975 CG89ET 73387745 IC50 > 20000 nM T88975 C3HSE2 73387863 IC50 > 20000 nM T88975 CU3D9N 73388373 IC50 = 50118.72 nM T88975 CHFG14 73425856 IC50 = 7840 nM T88975 C74TSX 73425972 IC50 = 7070 nM T88975 CWX3M6 73425973 IC50 = 16500 nM T88975 CEH2R6 73425974 IC50 = 4940 nM T88975 CK5SA7 73425975 IC50 = 7850 nM T88975 CRJ8D4 90665374 IC50 = 123000 nM T88975 CG5HV8 90668361 IC50 = 18700 nM T88975 C2HQ7I 90668362 IC50 = 29000 nM T88975 CDB74T 90668364 IC50 = 1500 nM T88975 C45QVJ 91668196 IC50 = 1600 nM T88975 CSCY01 117949009 IC50 = 8100 nM T88975 CXD39Z 118170767 IC50 = 10000 nM T88975 CYQ74R 118479645 IC50 > 10000 nM T88975 CM6XW1 118724093 IC50 = 29 nM T88975 C46LFG 118724094 IC50 = 37 nM T88975 CYM21X 118724095 IC50 = 17 nM T88975 C5TL8H 118725359 IC50 = 3700 nM T88975 CE49ML 118725368 IC50 = 167000 nM T88975 C4HI1Q 118729758 IC50 = 3300 nM T88975 CKBG19 118729759 IC50 = 1300 nM T88975 CRJE23 122185011 IC50 > 30000 nM T88975 CG0UN9 122189478 IC50 = 8150 nM T88975 CU1IF5 122189479 IC50 = 2990 nM T88975 CFK6E7 122189480 IC50 = 2450 nM T88975 CF18RV 122189481 IC50 = 3620 nM T88975 CFX0G3 122189482 IC50 = 240 nM T88975 COT7C8 122189483 IC50 = 1450 nM T88975 CD6AS1 122189484 IC50 = 1890 nM T88975 CLJ05T 122189485 IC50 = 6230 nM T88975 CJZ8X6 122189486 IC50 = 6890 nM T88975 CMDP54 122189487 IC50 = 7430 nM T88975 C0TXZ5 122189488 IC50 = 9120 nM T88975 CZTX23 122189489 IC50 = 9890 nM T88975 CH70PC 122189490 IC50 = 13440 nM T88975 CU2ZQ6 122189491 IC50 = 14630 nM T88975 CZW60O 122189492 IC50 = 16420 nM T88975 CJKO62 122193703 IC50 = 199000 nM T88975 C9W1JO 122193704 IC50 = 7710 nM T88975 C2MNX0 122193705 IC50 = 21900 nM T88975 C5EHB7 122193706 IC50 = 29500 nM T88975 C5WI6U 122193707 IC50 = 4070 nM T88975 COT0R6 122193708 IC50 = 22900 nM T88975 CJF36H 122193709 IC50 = 116000 nM T88975 C0J6MS 122193710 IC50 = 144400 nM T88975 C0XLR7 122193711 IC50 = 3740 nM T88975 CC9I0U 122193712 IC50 = 4510 nM T88975 CX30HD 122193713 IC50 = 25900 nM T88975 C6IJH8 122193928 IC50 = 3770 nM T88975 CNT17O 122193929 IC50 = 306000 nM T88975 C6Q5UO 122193930 IC50 = 66400 nM T88975 C1SWM0 122193931 IC50 = 62200 nM T88975 C9JSX0 122193932 IC50 = 58710 nM T88975 C6GI3B 122193933 IC50 = 78800 nM T88975 C9PTW4 122193934 IC50 = 810 nM T88975 C5FKM8 122193935 IC50 = 111000 nM T88975 C4UR7D 127038167 IC50 > 1000 nM T88975 C4H2TJ 127038168 IC50 > 1000 nM T88975 CL9JT8 127038169 IC50 > 1000 nM T88975 CJPX60 127038509 IC50 > 1000 nM T88975 C26EAG 127038511 IC50 > 1000 nM T88975 CTM9E4 127038512 IC50 > 1000 nM T88975 C6AQ2U 127038513 IC50 > 1000 nM T88975 CV1FM0 127038868 IC50 > 1000 nM T88975 CADU23 127038869 IC50 > 1000 nM T88975 CSY34W 127039587 IC50 > 10000 nM T88975 CACJ46 132489333 IC50 > 10000 nM T88975 CVA6W4 134147445 IC50 = 3.76 nM T88975 C1GY2T 135156251 EC50 > 10000 nM T88975 C3R8SE 135457869 IC50 > 10000 nM T88975 CJS37E 135482260 IC50 = 21900 nM T88975 C9IJK1 135566935 IC50 = 33200 nM T88975 C3PO9K 135856789 IC50 = 1890 nM T88975 CTX54Z 135896326 IC50 > 10000 nM T88975 C12UMG 136059728 IC50 > 1000 nM T88975 C8UF7G 136087052 IC50 > 50000 nM T88975 C21FVA 136180322 IC50 > 10000 nM T88975 C8TQ7A 136217455 IC50 > 50000 nM T88975 CH30RE 136260531 IC50 > 100000 nM T88975 CVG3Z1 136299192 IC50 = 1800 nM T88975 CRPN39 136645466 IC50 = 3200 nM T88975 CR53GQ 137290273 IC50 = 1800 nM T88975 C54KGS 137300710 IC50 = 750 nM T88975 C2N9VT 137348687 IC50 = 4200 nM T88975 CUKP61 137637556 IC50 = 3050 nM T88975 C9Q3PJ 137646307 IC50 = 3010 nM T88975 CQ3KH9 137650741 IC50 = 2750 nM T88975 CCVB31 137655787 IC50 = 2950 nM T88975 C6KYD7 137700754 IC50 > 10000 nM T88975 CM3UF7 137700779 IC50 > 20000 nM T88975 CPTE92 138319693 IC50 > 32000 nM T88975 CHJ79V 145997874 IC50 > 10000 nM T88975 CM7TX2 148279038 IC50 > 100000 nM T88975 CUT84A 155568798 IC50 > 100000 nM T88975 D06NIT 135564899 IC50 > 1000 nM T88975 D09RKU 46239428 Ki > 10000 nM T88975 D0H4UN 73211886 IC50 = 15000 nM T88975 D0J0CB 2753 IC50 = 16 nM T88975 D0R6MT 3758 IC50 = 7000 nM T50224 D0B5LF 448042 IC50 = 8300 nM T50224 D0EG1I 9926791 IC50 > 10000 nM T50224 D02ZQS 16095342 IC50 = 49 nM T50224 D03KKR 3547 IC50 = 5000 nM T50224 D0E3TC 44259 IC50 = 1.4 nM T50224 D0MS3Z 16725726 IC50 = 7940 nM T50224 D03BNU 59604787 IC50 > 10000 nM T50224 D0T3ME 156422 IC50 > 30000 nM T50224 C9VW8M 449054 IC50 > 16000 nM T50224 CP9AM1 599038 IC50 = 140 nM T50224 CJWX69 3848929 IC50 > 200000 nM T50224 CL5I2U 5330279 IC50 > 10000 nM T50224 CDK3J0 5703619 IC50 = 4 nM T50224 CM5Z8X 9869943 IC50 > 1000 nM T50224 CJO47T 9948405 IC50 > 10000 nM T50224 CV8I5X 9999342 IC50 > 10000 nM T50224 C1TQ7F 10171449 IC50 = 38 nM T50224 CUGP61 10214652 IC50 = 974 nM T50224 CWX0R6 10236187 IC50 = 17 nM T50224 C3TO7R 10236195 IC50 = 2120 nM T50224 CN3T7S 10236305 IC50 = 4390 nM T50224 C5TQ7X 10247543 IC50 > 10000 nM T50224 CRW7C6 10308125 IC50 = 1200 nM T50224 C5GTM6 10366534 IC50 > 10000 nM T50224 C2WQ8M 10473563 IC50 > 10000 nM T50224 CK63DE 10621161 IC50 = 4000 nM T50224 CRG03D 11245934 IC50 = 1000 nM T50224 C49NET 11256399 IC50 = 1 nM T50224 CKH0C4 11356881 IC50 = 20 nM T50224 C0APW4 11422034 IC50 = 10000 nM T50224 CACS26 11561968 Ki = 990 nM T50224 C5ER7L 11632412 IC50 = 4000 nM T50224 CKJ89S 11680113 IC50 = 126 nM T50224 CU0E8O 11690457 Ki = 94 nM T50224 CB0AP2 11705863 Ki > 1000 nM T50224 CHR92S 11858109 IC50 > 100000 nM T50224 C8E4TS 11992146 IC50 > 200000 nM T50224 CKR57M 16086104 IC50 > 25000 nM T50224 C16NRY 16086114 IC50 > 25000 nM T50224 C7Z4LV 16095343 IC50 = 14 nM T50224 CGC34R 16118737 IC50 > 100000 nM T50224 C54YXC 16121514 IC50 = 81.28 nM T50224 CUR7H3 16719862 IC50 = 146000 nM T50224 CHKM46 21590533 IC50 = 4000 nM T50224 CNKF46 21590534 IC50 = 4000 nM T50224 CG3VB6 23646578 IC50 = 3 nM T50224 CG6D4M 23647319 IC50 > 10000 nM T50224 CY8Z7X 23647330 IC50 > 10000 nM T50224 C4XD8H 23647348 IC50 > 10000 nM T50224 CDMI50 23661564 IC50 > 200000 nM T50224 CQNP54 24764449 IC50 = 100000 nM T50224 C4Z9CN 24769780 IC50 = 52000 nM T50224 CY8L7E 24896769 IC50 > 10000 nM T50224 CA9F3Y 25023714 IC50 = 21 nM T50224 C8Z4PI 25023715 IC50 = 15 nM T50224 CV96QX 25023716 IC50 = 3 nM T50224 C5INV4 25023717 IC50 = 47 nM T50224 CPOH02 25023718 IC50 = 11 nM T50224 C6F7RD 25023719 IC50 = 13 nM T50224 CPB4S2 25023721 IC50 = 162 nM T50224 C4DF8X 25023725 IC50 = 15850 nM T50224 C1JEU6 25023729 IC50 = 15800 nM T50224 CFH80B 25023733 IC50 = 10000 nM T50224 CR8JP7 25023735 IC50 = 8000 nM T50224 C4W7LY 25023736 IC50 = 19900 nM T50224 C0VQ1N 44396989 IC50 = 209 nM T50224 CE81DU 44396990 IC50 = 174 nM T50224 C70ZUC 44397010 IC50 = 1540 nM T50224 C18EWR 44397011 IC50 > 10000 nM T50224 C1W3CG 44397012 IC50 = 813 nM T50224 CCW02M 44397022 IC50 > 10000 nM T50224 C1N3EZ 44397032 IC50 = 3 nM T50224 C7M0VH 44397096 IC50 = 3 nM T50224 C62TNO 44397097 IC50 = 17 nM T50224 C0CST6 44397098 IC50 = 13 nM T50224 CDZA67 44397146 IC50 = 4 nM T50224 C3O4GA 44397147 IC50 = 229 nM T50224 C7YH8B 44397172 IC50 = 1520 nM T50224 C85BFL 44397176 IC50 = 10000 nM T50224 CCGI40 44397191 IC50 = 5097 nM T50224 CS5KW8 44397192 IC50 = 9 nM T50224 CNL87J 44397201 IC50 = 2240 nM T50224 CC3J1L 44397230 IC50 > 10000 nM T50224 CN2W1R 44397250 IC50 = 1.8 nM T50224 C2G1ME 44397259 IC50 = 7 nM T50224 CZY0I6 44397284 IC50 = 6 nM T50224 CL82EQ 44397285 IC50 = 8 nM T50224 C9QYL1 44397393 IC50 > 10000 nM T50224 CX68KE 44397418 IC50 > 10000 nM T50224 C8DZ7Q 44397421 IC50 = 55 nM T50224 CHR5J7 44397422 IC50 = 2.5 nM T50224 CU9J4N 44397451 IC50 = 13 nM T50224 C5QNX2 44397452 IC50 = 22 nM T50224 CI3S4C 44397453 IC50 = 4 nM T50224 CA1MH8 44397551 IC50 > 10000 nM T50224 C71TPW 44397578 IC50 = 9 nM T50224 C3WV9M 44397686 IC50 = 107 nM T50224 C18QWA 44397710 IC50 = 617 nM T50224 C47BPO 44397711 IC50 = 2 nM T50224 C3VRO9 44557921 IC50 > 10000 nM T50224 CLS29B 46872626 IC50 > 10000 nM T50224 C1NKE3 46905987 IC50 = 510 nM T50224 CJ2E9Q 46929857 IC50 > 25000 nM T50224 CHSF07 49806372 IC50 > 1000 nM T50224 CEQN27 52936621 Ki > 1000 nM T50224 C8NA4L 53384644 IC50 > 30000 nM T50224 CM8JX1 56604907 IC50 = 10000 nM T50224 C1MR8Q 60097495 IC50 > 10000 nM T50224 CV63UL 67240318 IC50 > 10000 nM T50224 C5D1LV 70687790 IC50 = 4570.88 nM T50224 C1IEJ2 70789254 IC50 = 5300 nM T50224 C8T7ZP 70789255 IC50 = 700 nM T50224 CE1QA0 135493216 IC50 = 258 nM T50224 CY4D8I 135566504 Ki = 728.5 nM T50224 CG3UZ1 135927974 Ki > 1000 nM T50224 CXS84F 136030409 IC50 = 1960 nM T50224 CAWR70 136109070 IC50 > 10000 nM T50224 C2MD1Q 155513187 IC50 > 10000 nM T50224 D00ERW 44444843 Ki > 1892 nM T50224 D03DZO 11715767 IC50 = 2340 nM T50224 D05GSF 44397277 IC50 = 1.4 nM T50224 D07OXC 11650194 IC50 > 100000 nM T50224 D09FFE 449241 IC50 = 120 nM T50224 D0EW9J 10389239 IC50 > 200000 nM T50224 D0I1FJ 11393719 IC50 = 0.5 nM T50224 D0M5FF 5083 IC50 = 8 nM T50224 D0OZ2S 11785878 IC50 > 100000 nM T14908 D0D0ZD 441314 IC50 > 1000000 nM T14908 D0HR8Z 51634 IC50 = 20000 nM T14908 D0MU9L 176077 IC50 > 100000 nM T14908 D0RE9C 501391 IC50 = 10000 nM T14908 D0S5LT 29435 IC50 > 100000 nM T14908 C1EH0P 501640 IC50 = 1600 nM T14908 CG2I5E 6610216 IC50 = 23000 nM T14908 CC7F5J 9929494 IC50 = 4000 nM T14908 C3O2JI 10093000 IC50 = 1000 nM T14908 CAWL97 10888248 IC50 = 9000 nM T14908 C06FUY 11105683 IC50 > 100000 nM T14908 CC4N0X 11258014 IC50 = 100 nM T14908 C1UV7P 11406578 IC50 = 164000 nM T14908 C5MYQ2 11569854 IC50 = 90 nM T14908 CYS8W0 11648559 IC50 = 90 nM T14908 C1JBA9 11816841 IC50 > 100000 nM T14908 CZ21NH 23622616 IC50 = 10000 nM T14908 C1RDO2 23652731 IC50 = 16 nM T14908 CWF97M 23652732 IC50 = 9 nM T14908 CQ3SX9 44820249 IC50 = 500 nM T14908 CNL06X 44820252 IC50 > 100000 nM T14908 CO1BZ7 46847258 IC50 = 10 nM T14908 CXFW51 46850909 IC50 = 32 nM T14908 CP9LO1 46868871 IC50 = 2 nM T14908 CH60VD 46868943 IC50 = 230 nM T14908 CDG7J2 46868944 IC50 = 2 nM T14908 CA65DY 46869010 IC50 = 1075 nM T14908 C0YU3X 46869012 IC50 = 1080 nM T14908 CV0C3Y 46869239 IC50 = 7 nM T14908 CB64IV 46869370 IC50 = 180 nM T14908 CO0ID6 46869371 IC50 = 3 nM T14908 CPHL15 46869372 IC50 = 90 nM T14908 CS18VL 46869438 IC50 = 110 nM T14908 CO7N4V 46869440 IC50 = 50 nM T14908 CV8U0E 46869507 IC50 = 340 nM T14908 CFS4H5 46869564 IC50 = 2700 nM T14908 C56YTJ 46869566 IC50 = 120 nM T14908 C4XSW2 46869622 IC50 = 1150 nM T14908 C4OTC7 46869623 IC50 = 53 nM T14908 CKH9U1 46869624 IC50 = 300 nM T14908 C0LRS2 46869760 IC50 = 275 nM T14908 CQR58G 46892601 IC50 = 20 nM T14908 CIX16G 46892972 IC50 = 90 nM T14908 CK6Z7P 46892975 IC50 = 160 nM T14908 CS4XV6 46892977 IC50 = 3 nM T14908 C98JRZ 46893358 IC50 = 7 nM T14908 CDVO63 56928630 IC50 = 5 nM T14908 C9OLQ7 57392788 IC50 = 20 nM T14908 C6KF4Q 57394510 IC50 = 2 nM T14908 CCEO27 57394520 IC50 = 1 nM T14908 C65DMS 57398065 IC50 = 10 nM T14908 CCS9O0 57398066 IC50 = 4 nM T14908 CIOZ69 57399724 IC50 = 2 nM T14908 C3JYL4 57403223 IC50 = 9 nM T14908 CSL60R 57403230 IC50 = 50 nM T14908 C78GME 57403231 IC50 = 40 nM T14908 CU5J8W 57403232 IC50 = 65 nM T14908 CKVH81 57403233 IC50 = 7 nM T14908 C3VL6I 57522017 IC50 = 2 nM T14908 CBC85H 57522018 IC50 = 4 nM T14908 CIK6G9 57522019 IC50 = 150 nM T14908 CW23VX 57522130 IC50 = 190 nM T14908 CT13YK 57522131 IC50 = 2 nM T14908 C20IFP 57522132 IC50 = 4 nM T14908 CW50IU 57522133 IC50 = 260 nM T14908 C6E5BW 57522134 IC50 = 3 nM T14908 C43URP 57522135 IC50 = 16 nM T14908 CYU9J7 57522248 IC50 = 2 nM T14908 CWLD45 57522249 IC50 = 3 nM T14908 C2K5MR 57522250 IC50 = 3 nM T14908 C6HTG0 57522251 IC50 = 2 nM T14908 C13WLT 57522252 IC50 > 4000 nM T14908 C2NXA4 101882899 IC50 = 60 nM T14908 C05DUA 101882900 IC50 = 2.5 nM T14908 CU1NL5 118411065 IC50 = 100 nM T14908 CH5U7F 118411068 IC50 = 25 nM T14908 C8X6RN 118411069 IC50 = 5 nM T14908 C16QGB 118411070 IC50 = 8 nM T14908 CD76NI 118411071 IC50 = 25 nM T14908 C9LGB3 118411072 IC50 = 25 nM T14908 CAR82K 118411073 IC50 = 50 nM T14908 CGXZ37 118411074 IC50 = 25 nM T14908 C8G3LO 118411076 IC50 = 50 nM T14908 CB72ZY 118411077 IC50 = 1250 nM T14908 C97IKP 118411079 IC50 = 2000 nM T14908 CV78UK 118411080 IC50 = 200 nM T14908 CC84LW 118411081 IC50 = 150 nM T14908 C2CF0W 118411108 IC50 = 3 nM T14908 C89IWU 118411135 IC50 = 50 nM T14908 C5PIW8 118411136 IC50 = 150 nM T14908 CY83DV 118411140 IC50 = 100 nM T14908 CFH4O0 118411147 IC50 = 150 nM T14908 CH7BA2 118411149 IC50 = 3 nM T14908 CUYO63 118411153 IC50 = 25 nM T14908 CMB63J 118719880 IC50 = 500 nM T14908 C5N8JX 118719882 IC50 = 300 nM T14908 CL6Y0C 118719883 IC50 = 1000 nM T14908 C53BCZ 118719884 IC50 = 300 nM T14908 CP0E3J 118719886 IC50 = 750 nM T14908 C8EXK9 118719887 IC50 = 3 nM T14908 CN6TK0 118719889 IC50 = 3 nM T14908 CL97RN 118719890 IC50 = 70 nM T14908 C60DKA 118719891 IC50 = 400 nM T14908 C5HZB0 118719893 IC50 = 250 nM T14908 C6OML9 118719895 IC50 = 1000 nM T14908 C1P9FV 118719896 IC50 = 80 nM T14908 C86SLH 118719897 IC50 = 2500 nM T14908 CDTA82 118719898 IC50 = 200 nM T14908 CXOU16 118719899 IC50 = 3 nM T14908 CD56OM 118719901 IC50 = 3 nM T14908 C3WIV2 118719902 IC50 = 100 nM T14908 CI1OS6 118719903 IC50 = 25 nM T14908 CSTV68 118719904 IC50 = 25 nM T14908 CX4WV8 118719905 IC50 = 150 nM T14908 C1D3IO 118719906 IC50 = 50 nM T14908 CPVS50 118719907 IC50 = 25 nM T14908 CP9E1B 118719908 IC50 = 25 nM T14908 CHP35O 118719909 IC50 = 75 nM T14908 CZC89F 118719910 IC50 = 25 nM T14908 CE72DG 118719911 IC50 = 20 nM T14908 CCU4F2 118719912 IC50 = 20 nM T14908 CZ0PY7 118719913 IC50 = 25 nM T14908 C5JQ8G 118719914 IC50 = 40 nM T14908 C1MGA5 118719915 IC50 = 25 nM T14908 CT6GP0 118719916 IC50 = 2000 nM T14908 C1SJU6 118719917 IC50 = 2000 nM T14908 CR67QX 118719918 IC50 = 750 nM T14908 CC8N6I 118719919 IC50 = 75 nM T14908 C1WON3 118720302 IC50 = 70 nM T14908 C0ZOT7 118720303 IC50 = 60 nM T14908 C81YUI 118720304 IC50 = 40 nM T14908 CXI04D 118720305 IC50 = 30 nM T14908 CG7JV9 118720306 IC50 = 70 nM T14908 CR4S5Y 118720307 IC50 = 20 nM T14908 CG9Q8E 118720308 IC50 = 15 nM T14908 D0N9IX 9822159 IC50 = 90 nM T55959 D01AXB 60835 Ki = 240 nM T55959 D01JMC 11658860 Ki > 10000 nM T55959 D01UTL 2995 Ki = 0.49 nM T55959 D02PPN 4158 IC50 = 17 nM T55959 D02XOK 6917779 IC50 = 3200 nM T55959 D03HFG 5324346 Ki = 1.46 nM T55959 D04CRN 54841 IC50 = 3100 nM T55959 D04XPW 446220 Ki = 32 nM T55959 D06GDY 43815 Ki = 400 nM T55959 D06ZUK 3696 IC50 = 25600 nM T55959 D07HQC 4236 Ki = 927 nM T55959 D09VGC 65833 IC50 > 10000 nM T55959 D0CQ0Z 33630 Ki = 1714 nM T55959 D0H8QL 4020 IC50 = 13 nM T55959 D0HQ6N 1201549 IC50 = 312 nM T55959 D0J5RN 9690109 Ki = 647 nM T55959 D0K0TC 68617 IC50 = 310 nM T55959 D0O3FG 125017 Ki > 854 nM T55959 D0P1UX 5656 Ki > 890 nM T55959 D0T3LF 5826 EC50 = 24.8 nM T55959 D0T7OW 681 IC50 = 460 nM T55959 D0TR5X 3386 Ki = 1900 nM T55959 D0X4ZR 444 Ki = 441 nM T55959 D0Y5DO 2771 Ki = 16540 nM T55959 D0Y5UG 2160 Ki = 6203 nM T55959 D0ZS8P 2801 IC50 = 2777 nM T55959 D00JFE 56941241 IC50 = 3400 nM T55959 D00WLO 3455 Ki = 0.36 nM T55959 D03QIE 47953 IC50 = 910 nM T55959 D04PXS 11658655 Ki = 79.43 nM T55959 D07AHC 65650 IC50 = 1300 nM T55959 D0F5NJ 1615 Ki = 897 nM T55959 D0J9PT 58212050 IC50 = 5.7 nM T55959 D0LI1C 44469321 IC50 > 10000 nM T55959 D0R2OU 25070031 IC50 = 9400 nM T55959 D0WL3H 15983287 IC50 = 491 nM T55959 D08DMM 91799365 IC50 = 730 nM T55959 D0LI2I 118096900 IC50 > 10000 nM T55959 D0QE8S 60197821 IC50 = 1380 nM T55959 D01NJT 65856 Ki > 2000 nM T55959 D06BPG 4528 Ki = 10 nM T55959 D08AWI 11430856 Ki > 2000 nM T55959 D0A5RD 9795056 IC50 = 220 nM T55959 D0G1RH 6918446 IC50 = 0.2 nM T55959 D0H9GQ 9795276 IC50 = 78 nM T55959 CLJ8R2 1576 EC50 = 12.5 nM T55959 C6YZ2N 8554 IC50 > 100000 nM T55959 CK9A6Z 9280 IC50 = 19.9 nM T55959 C5H9CN 9287 Ki = 666 nM T55959 CRU9X7 16458 Ki > 10000 nM T55959 C3VL1J 27694 Ki > 10000000 nM T55959 C3L9YO 36663 Ki = 5700 nM T55959 CGU3Z5 42145 Ki = 8510 nM T55959 CQR7U2 44024 Ki = 7.2 nM T55959 C1JV7L 52940 Ki = 17 nM T55959 C0OST7 55993 Ki = 7 nM T55959 C6KXM1 62857 IC50 = 18400 nM T55959 C9E6LD 62923 IC50 = 15700 nM T55959 CI6QK3 77250 Ki = 742 nM T55959 C8X5YU 77251 Ki = 780 nM T55959 C0O3IG 77252 Ki = 79 nM T55959 CYKE31 104920 Ki = 2.42 nM T55959 C5Q1OD 108220 Ki = 6.34 nM T55959 CH0S2U 125416 Ki = 32.36 nM T55959 CXUG79 148883 IC50 > 10000 nM T55959 CZ1C9K 154101 Ki = 16 nM T55959 CBJ51L 190851 Ki = 13.49 nM T55959 CD1H4C 204666 IC50 = 730 nM T55959 C28RMF 214398 IC50 = 110 nM T55959 CQ97NL 242919 Ki = 99 nM T55959 C1KUD9 264388 Ki > 10000 nM T55959 CR7MP9 264389 Ki > 10000 nM T55959 CQK09D 279413 Ki = 390 nM T55959 CR92BY 285225 IC50 = 548 nM T55959 CT9SV0 403506 IC50 = 67.1 nM T55959 CAMF37 403507 IC50 = 359 nM T55959 CDR63W 403508 Ki = 2.83 nM T55959 CE3N8G 411735 Ki = 2731 nM T55959 C97TAX 516222 IC50 = 3600 nM T55959 CZ53QF 656832 Ki = 46.3 nM T55959 CZN6S9 743974 IC50 > 100000 nM T55959 C2CT0Y 818024 Ki = 115 nM T55959 CK65MQ 826771 IC50 = 9900 nM T55959 CO2SD9 1076689 IC50 = 1700 nM T55959 CQ0DV9 1393540 IC50 = 16000 nM T55959 C47BIF 1394484 IC50 = 675 nM T55959 CH24PD 2801930 Ki = 969 nM T55959 CA3S7R 3022645 Ki = 60 nM T55959 CZ9SV5 3025846 Ki = 1.1 nM T55959 CK8F0T 3080846 IC50 = 95 nM T55959 C9HJ3S 3302814 Ki = 2038 nM T55959 C0YXV3 3676358 Ki > 10000 nM T55959 CF12IO 4141883 Ki = 371 nM T55959 COC2V5 4913097 IC50 = 980 nM T55959 CI56AJ 5141361 Ki = 0.69 nM T55959 C5FUA2 6328322 Ki = 17400 nM T55959 C8ZK1O 6328354 Ki = 7.2 nM T55959 C0IHP9 6336338 Ki = 23.5 nM T55959 CY70ST 9794826 IC50 > 10000 nM T55959 C2ICW4 9794964 Ki = 10.6 nM T55959 CDEL49 9795462 Ki = 40.5 nM T55959 C6XYV0 9795623 IC50 = 19600 nM T55959 CR2JV1 9795977 Ki = 77 nM T55959 CY86MJ 9796441 IC50 = 17 nM T55959 C65YOK 9797476 Ki = 6.31 nM T55959 C5FJ4K 9798438 IC50 = 170 nM T55959 CZGK19 9801045 Ki = 263.03 nM T55959 C8XGV3 9804849 IC50 = 10000 nM T55959 C15SGM 9814918 IC50 = 286 nM T55959 C7PUZ1 9816962 Ki = 78 nM T55959 CT7OD0 9817610 Ki > 200 nM T55959 CB8N5S 9817852 IC50 = 0.83 nM T55959 CEPW14 9834659 IC50 = 44000 nM T55959 CQPO85 9835750 IC50 = 3.1 nM T55959 C05OSH 9836383 Ki = 14 nM T55959 CM85OH 9836429 IC50 = 14 nM T55959 C3DN1P 9836520 IC50 = 3.3 nM T55959 CX8P7C 9837869 Ki = 233 nM T55959 CAL4C9 9837874 IC50 = 3 nM T55959 CY7K5Z 9838051 Ki = 98.8 nM T55959 C1YLP0 9838350 Ki = 36 nM T55959 C0YI3N 9839972 IC50 = 370 nM T55959 C43EZB 9857586 IC50 = 736 nM T55959 C7D0UC 9861237 IC50 = 29.1 nM T55959 CIXO17 9863396 Ki = 1.05 nM T55959 C0IR5C 9864943 Ki = 370 nM T55959 C1ZB4W 9865652 Ki > 1000 nM T55959 C3KGX7 9867350 Ki = 210 nM T55959 CN9YD5 9868131 IC50 = 200 nM T55959 CQ4LC2 9872676 Ki = 1800 nM T55959 CEJP40 9878793 IC50 = 707 nM T55959 C01ABG 9881528 Ki = 61 nM T55959 CCZ84V 9881969 Ki = 106 nM T55959 CT6C5H 9881970 Ki = 58 nM T55959 CHNC28 9882029 Ki = 64 nM T55959 CY6QX4 9882047 Ki = 44.7 nM T55959 C7KP4G 9882069 Ki = 12893 nM T55959 CQ2BS0 9884087 IC50 = 6500 nM T55959 C8Q4OZ 9884474 Ki = 8.7 nM T55959 CBQ7Y3 9886288 Ki > 1000 nM T55959 CN52BU 9887951 IC50 = 1500 nM T55959 CM3L0I 9900725 IC50 = 2630 nM T55959 CZUM05 9900755 IC50 = 27 nM T55959 CCFR97 9903806 Ki = 18 nM T55959 CPH07N 9903956 Ki = 21.5 nM T55959 CYWQ50 9906447 Ki > 10000 nM T55959 CUEZ75 9908121 IC50 = 2.9 nM T55959 CCM2Z0 9908126 IC50 = 90 nM T55959 C1CSK2 9910220 IC50 = 0.37 nM T55959 CSKJ62 9910492 IC50 = 100 nM T55959 CL5W7J 9920766 IC50 > 100000 nM T55959 CQX6R9 9924713 IC50 > 10000 nM T55959 C3RVK7 9928961 IC50 = 450 nM T55959 C10VOI 9930235 IC50 = 1100 nM T55959 CPYN79 9930791 IC50 = 270 nM T55959 C6AZ3X 9943908 IC50 = 1600 nM T55959 C7QFK2 9947230 IC50 = 0.4 nM T55959 CPBQ94 9948049 IC50 = 5270 nM T55959 CK65YF 9948112 Ki = 0.22 nM T55959 CM7J6H 9948700 IC50 = 12 nM T55959 CAP9K6 9949231 IC50 = 1.16 nM T55959 C76NBU 9950374 Ki > 10000 nM T55959 C5JI4O 9951619 IC50 = 270 nM T55959 C79VHZ 9952054 IC50 = 1.26 nM T55959 CMI58L 9956563 IC50 = 0.059 nM T55959 CFZ9D7 9972515 IC50 = 2 nM T55959 COP08X 9972881 IC50 = 4.8 nM T55959 CD8T5E 9976807 Ki = 23.44 nM T55959 CXCP15 9980795 IC50 = 47 nM T55959 C2AW8E 9996581 Ki = 0.2 nM T55959 CJ95XF 10003490 Ki = 30 nM T55959 CD9JO4 10015148 IC50 = 660 nM T55959 CHG91I 10017115 Ki > 10000 nM T55959 CD6B7Q 10025195 IC50 = 35 nM T55959 CL06BD 10027543 Ki = 4.4 nM T55959 C3Z4OD 10040286 Ki > 10000 nM T55959 C25WVJ 10047566 IC50 > 1000 nM T55959 C86EDS 10048368 Ki = 28.18 nM T55959 C5MQ9L 10060174 IC50 = 67 nM T55959 COZ94V 10062443 Ki = 962 nM T55959 C79GJK 10062560 Ki > 2000 nM T55959 C1J4YU 10072978 Ki = 90 nM T55959 C5HJ1G 10073022 Ki = 38.9 nM T55959 CKY83M 10078142 IC50 = 18 nM T55959 C1LN4V 10084648 IC50 > 100 nM T55959 CO50KM 10085525 Ki = 2651 nM T55959 C6L5KD 10086762 IC50 = 7.1 nM T55959 CW7K1U 10086952 Ki = 163500 nM T55959 C5H3MJ 10090352 IC50 = 6 nM T55959 CPQD23 10096087 Ki = 3 nM T55959 CO1R2Q 10110820 IC50 > 10000 nM T55959 CINW17 10130931 Ki = 112 nM T55959 C80GWE 10132137 IC50 = 7.37 nM T55959 C4BS0C 10189446 IC50 = 10 nM T55959 C13VPI 10198613 Ki = 276 nM T55959 CM9CT0 10198980 Ki = 36 nM T55959 C4J6DM 10199240 Ki = 25 nM T55959 CF9B2N 10220613 Ki = 27 nM T55959 CG32IU 10220615 Ki = 227 nM T55959 CI8NQ2 10220697 Ki = 30.1 nM T55959 C8C6IY 10221010 IC50 = 690 nM T55959 C6HUY5 10238982 Ki = 1.3 nM T55959 C2D4YM 10244152 IC50 > 100 nM T55959 CMSE68 10245407 IC50 = 89 nM T55959 CQ4M3F 10265481 Ki > 10000 nM T55959 C5AX7N 10291757 Ki = 309 nM T55959 C5HI6T 10293752 IC50 = 8000 nM T55959 CB4C9E 10313840 Ki > 5000 nM T55959 C1Z8AO 10314993 Ki = 53 nM T55959 CKE53N 10320283 IC50 = 1070 nM T55959 CUF4G8 10355130 Ki = 38 nM T55959 CLG82T 10356463 Ki > 10000 nM T55959 CK1X4I 10356972 IC50 = 2 nM T55959 C1A0VI 10359867 Ki = 0.67 nM T55959 CRZ15J 10363398 Ki = 3.5 nM T55959 C3R7VI 10367506 Ki = 0.71 nM T55959 CN1L4S 10377587 IC50 = 750 nM T55959 CX13CN 10381502 Ki = 45 nM T55959 CN2O8Q 10400315 Ki = 279 nM T55959 CEAN45 10402966 IC50 = 2.9 nM T55959 C23LGF 10411109 Ki = 18 nM T55959 C2B0IU 10421236 Ki = 2350 nM T55959 CV7H9G 10424170 Ki = 501.19 nM T55959 CI9ZQ8 10428183 IC50 = 44 nM T55959 CL0ZB2 10430935 Ki = 720 nM T55959 CR8J7I 10432519 Ki = 17 nM T55959 CRKC54 10439429 Ki = 6.7 nM T55959 C98SIQ 10446567 Ki > 1000 nM T55959 CL65VJ 10450883 Ki = 5.25 nM T55959 C5Q2IO 10472386 Ki = 3.2 nM T55959 CSZ56B 10472714 IC50 = 1.09 nM T55959 C5HDQ3 10476240 IC50 = 30 nM T55959 C86GXB 10477812 Ki = 2.3 nM T55959 CT9IP1 10477960 Ki = 10.9 nM T55959 CRZ59G 10479666 Ki = 0.75 nM T55959 C8UYW6 10494535 Ki = 501.19 nM T55959 C7G9HB 10499540 Ki = 25.7 nM T55959 C5MGB6 10503847 Ki = 371.54 nM T55959 CF7B1H 10520686 Ki = 130 nM T55959 COML53 10521074 Ki = 3.236 nM T55959 CX69HP 10525046 Ki = 83 nM T55959 C7GHM2 10525660 Ki = 114.82 nM T55959 CXJ4S9 10527655 Ki = 371.54 nM T55959 C7TX6Q 10543664 Ki = 530 nM T55959 CJ6P1Z 10544672 Ki = 250 nM T55959 C3DR1F 10551367 Ki = 87 nM T55959 CP1RV2 10551946 Ki = 41.69 nM T55959 C0US7T 10568696 Ki = 680 nM T55959 COA6T3 10570967 IC50 = 1 nM T55959 C4FAY9 10574379 Ki = 15.14 nM T55959 C4U6NW 10575012 Ki = 61 nM T55959 C3CYF7 10575547 IC50 > 10 nM T55959 CC12NB 10591764 Ki = 32 nM T55959 CNB16D 10593212 Ki = 0.6761 nM T55959 CZT6V3 10598567 Ki = 501.19 nM T55959 CAGB14 10598649 Ki = 160 nM T55959 CZ6HL3 10600622 Ki = 93.33 nM T55959 CQW4H8 10627068 Ki = 26 nM T55959 C8L4AG 10640435 Ki = 180 nM T55959 C69FME 10640436 Ki = 1000 nM T55959 C71KTR 10645578 IC50 = 3213 nM T55959 C6ZF8N 10657292 IC50 = 1200 nM T55959 CCZU47 10663468 Ki = 39 nM T55959 C91PBZ 10663685 Ki = 47.86 nM T55959 C2P5WV 10666153 Ki = 323 nM T55959 CQ7V9F 10670209 IC50 > 10 nM T55959 CX12VM 10670307 Ki = 122 nM T55959 C0VWZ3 10672803 IC50 = 33 nM T55959 C5FY3Q 10688125 Ki = 650 nM T55959 CU58VP 10691286 Ki = 120 nM T55959 CG0V7W 10693838 Ki = 210 nM T55959 CTS2I1 10696077 Ki = 28.84 nM T55959 CRLX06 10697639 Ki = 1.72 nM T55959 C26VWI 10712698 Ki = 890 nM T55959 C2SK7H 10716649 Ki = 501.19 nM T55959 CPO3J8 10734429 Ki = 450 nM T55959 CP5DO8 10739933 IC50 = 37.6 nM T55959 C3I7ZE 10740824 Ki = 30 nM T55959 CDZT46 10741033 Ki = 16.98 nM T55959 CRP3D6 10765459 Ki = 51 nM T55959 C1RA7B 10786304 Ki = 112.2 nM T55959 CP1N4Y 10788455 Ki = 54 nM T55959 CGM3Q2 10788465 Ki = 28 nM T55959 CUV46I 10810932 Ki = 46.77 nM T55959 C2Q4BI 10813108 Ki = 70 nM T55959 CNB26G 10813109 IC50 = 210 nM T55959 C1C5KZ 10835318 Ki = 14.13 nM T55959 C9M7UN 10835740 Ki = 322 nM T55959 C0GX8V 10836499 Ki = 110 nM T55959 C1GAE4 10837110 Ki = 100 nM T55959 C83QOV 10851850 Ki = 501.19 nM T55959 CAM8P0 10852732 Ki = 64 nM T55959 C5JU4D 10860718 IC50 = 2.7 nM T55959 CRI50E 10885636 IC50 = 996 nM T55959 CP42DJ 10891958 IC50 = 146 nM T55959 CMS0Z2 10893018 IC50 = 10.6 nM T55959 CY9RE6 10894733 Ki = 34.67 nM T55959 C1AU9X 10895029 Ki = 10.96 nM T55959 C58SAQ 10904197 Ki = 2.01 nM T55959 CWJL70 10905740 IC50 = 1520 nM T55959 CX65PW 10907460 IC50 = 994 nM T55959 CLP15C 10911476 IC50 = 13000 nM T55959 CE9JL7 10934835 IC50 = 59 nM T55959 C9VH4C 10946580 Ki = 698 nM T55959 CUG82R 10993971 Ki = 5.3 nM T55959 C15TXK 10994187 Ki = 0.73 nM T55959 C9VHZ5 11000971 IC50 = 125 nM T55959 CI6XZ2 11001331 IC50 = 1260 nM T55959 CJC9K4 11005810 IC50 = 781 nM T55959 CSD70W 11033919 IC50 = 1841 nM T55959 CW0B4J 11034392 Ki = 10.3 nM T55959 CEK01S 11044358 IC50 > 100000 nM T55959 CZ35QF 11045269 Ki = 6 nM T55959 CN4A0J 11046488 Ki = 18.2 nM T55959 C6EBF3 11048769 IC50 = 2940 nM T55959 C2ZB0J 11059071 Ki = 25 nM T55959 CG41BK 11071079 IC50 = 1650 nM T55959 C3XW2P 11077246 IC50 = 30.4 nM T55959 CIL61D 11077445 IC50 = 4.1 nM T55959 C19OWN 11088955 IC50 = 218 nM T55959 CIE70M 11089063 IC50 = 8.4 nM T55959 C9KZ6L 11091998 Ki = 1.61 nM T55959 CUR50W 11098085 IC50 = 4000 nM T55959 CV1TH4 11102046 Ki = 30.9 nM T55959 CXNV12 11102187 Ki = 0.99 nM T55959 C2IN5D 11102683 Ki = 12 nM T55959 C7DE0U 11113605 IC50 = 1280 nM T55959 C2ALP4 11130459 IC50 = 12.3 nM T55959 CR6J8C 11130848 Ki = 2.9 nM T55959 CW49ZY 11132158 IC50 = 390 nM T55959 CLRV35 11134191 Ki = 1.3 nM T55959 C5SP9Y 11139047 IC50 = 3000 nM T55959 C8W5NR 11145001 Ki = 1.01 nM T55959 C36VJK 11149970 Ki = 2121 nM T55959 CT7Z9R 11150712 Ki = 275 nM T55959 C39INR 11150726 Ki = 11.5 nM T55959 CP7O3X 11161917 Ki = 2908 nM T55959 CKB2H1 11163292 IC50 = 4.5 nM T55959 CK27CU 11164446 Ki > 1000 nM T55959 C95YLA 11173366 Ki = 1960 nM T55959 C7OEX0 11174494 Ki = 430 nM T55959 CLE8G5 11176087 Ki = 309 nM T55959 CAN73X 11189693 IC50 = 500 nM T55959 CM1T4L 11197267 Ki = 105 nM T55959 CXQ48K 11198677 IC50 = 389 nM T55959 CPX23W 11209208 Ki = 460 nM T55959 CPH9Q8 11210071 IC50 > 6000 nM T55959 CJ0K8E 11213696 Ki = 5.012 nM T55959 C3VT2W 11219249 IC50 = 42 nM T55959 CCR0V5 11224454 Ki = 4426 nM T55959 CA39QR 11227406 Ki = 490 nM T55959 CR7IZ6 11231488 Ki = 28.8 nM T55959 CPVA01 11255359 IC50 = 0.75 nM T55959 C6IRX4 11265803 Ki > 1000 nM T55959 CG4R6Y 11266831 Ki > 200 nM T55959 C9S3BR 11267769 IC50 = 9.1 nM T55959 C6A0RY 11276613 Ki = 5296 nM T55959 C27GXZ 11277680 Ki = 30.2 nM T55959 CXH8G3 11278436 IC50 = 6.4 nM T55959 CG9TM7 11293593 Ki > 10000 nM T55959 C57GTA 11299968 IC50 = 283 nM T55959 CP26RV 11300496 Ki = 1330 nM T55959 C3F7NY 11301501 IC50 > 40000 nM T55959 CKQ7E8 11301538 Ki > 5000 nM T55959 CV1LG4 11301893 IC50 > 4000 nM T55959 CP12MY 11302314 IC50 = 212 nM T55959 CS3BL0 11310988 Ki = 2100 nM T55959 CUXZ91 11311148 IC50 = 16.3 nM T55959 C2GZD3 11311204 IC50 = 49.7 nM T55959 CCJA60 11323414 Ki = 1610 nM T55959 CBA4U5 11335494 IC50 = 18.3 nM T55959 CF2X6Y 11336016 Ki = 2400 nM T55959 CH83FN 11346324 Ki > 1000 nM T55959 CXZ82E 11347860 Ki = 135 nM T55959 C3O0EP 11349976 Ki = 340 nM T55959 C4ZP2J 11358065 IC50 = 27 nM T55959 C8J5NW 11361155 IC50 = 6.7 nM T55959 CR5S4A 11368527 IC50 = 55 nM T55959 C7MN8V 11391287 IC50 = 5.9 nM T55959 CE85CL 11415039 IC50 = 154 nM T55959 CE2TS1 11425104 Ki = 1330 nM T55959 CU4H7W 11426687 Ki > 10000 nM T55959 C85LYP 11430418 IC50 > 1000 nM T55959 C6E3VO 11449834 Ki = 144 nM T55959 CMH9J5 11450298 IC50 = 89 nM T55959 CX3ZU0 11450539 IC50 > 4000 nM T55959 CNS8J9 11459667 IC50 = 44.3 nM T55959 CF5R1Z 11463970 IC50 = 3.9 nM T55959 C9L2AH 11474847 IC50 = 11 nM T55959 C2X3OY 11483535 Ki > 5000 nM T55959 CZ7X9M 11492164 IC50 > 10000 nM T55959 C7G5HP 11492305 IC50 > 10000 nM T55959 CA8KE0 11492902 IC50 = 1500 nM T55959 C3XD4T 11493035 Ki > 10000 nM T55959 C2NJY3 11499666 IC50 = 18680 nM T55959 C2X7HI 11499753 Ki > 10000 nM T55959 C7UJM8 11499957 IC50 = 8.6 nM T55959 CDC5I4 11499958 Ki = 3.7 nM T55959 CXR70Z 11500795 Ki = 3960 nM T55959 C3B0LO 11501191 Ki > 10000 nM T55959 CR1K9A 11504964 Ki = 1.3 nM T55959 C2Y0JA 11505593 Ki = 12 nM T55959 CS1YI5 11506975 IC50 > 10000 nM T55959 C9OV2L 11507416 IC50 = 200 nM T55959 C6FA1G 11513575 Ki = 18 nM T55959 CM3P5D 11514441 Ki > 10000 nM T55959 C9XYF3 11521964 IC50 = 231 nM T55959 C75FPD 11529874 Ki = 3740 nM T55959 C38QFE 11530118 Ki > 10000 nM T55959 C6SCW7 11536158 Ki = 34790 nM T55959 CQ08DH 11539632 IC50 > 10 nM T55959 CC67XR 11543737 IC50 = 266 nM T55959 CGV24I 11544186 IC50 = 1120 nM T55959 CWCU85 11548538 Ki = 1.7 nM T55959 CTXP63 11550888 IC50 = 38 nM T55959 C9VC7O 11551780 Ki = 8440 nM T55959 C3RMI1 11559300 Ki = 3570 nM T55959 CY71DQ 11562044 Ki = 1.4 nM T55959 C1VF0P 11566266 Ki > 10000 nM T55959 CDP9Z0 11566316 Ki = 3040 nM T55959 C8C1VW 11566318 Ki = 4770 nM T55959 CIE3O7 11566487 Ki = 1530 nM T55959 CZD62R 11572546 IC50 > 12000 nM T55959 CMX60P 11573849 IC50 = 5870 nM T55959 C6JC2T 11580039 Ki > 10000 nM T55959 C2T6RF 11584839 Ki = 0.9 nM T55959 CMZ54K 11587069 Ki = 6500 nM T55959 C3LAI9 11587242 IC50 = 53 nM T55959 CY3A4K 11587772 Ki = 2950 nM T55959 CU8F6B 11588595 IC50 = 570 nM T55959 CI12ZR 11592176 Ki = 1.1 nM T55959 CW1CO6 11594137 IC50 = 44 nM T55959 CZ6US0 11594677 IC50 = 11.8 nM T55959 CJ27XH 11594827 Ki > 4000 nM T55959 CAD20M 11598831 Ki = 1.4 nM T55959 C9YR3G 11599258 Ki = 1.4 nM T55959 C7UFA1 11600778 IC50 > 10000 nM T55959 CE4GZ0 11609767 Ki = 520 nM T55959 C6HLN8 11610150 Ki = 4650 nM T55959 C8JAM4 11616357 IC50 = 339 nM T55959 CCM6U9 11616771 Ki = 2610 nM T55959 C1F4DL 11618807 Ki = 46 nM T55959 CXR9Y6 11619798 Ki = 253 nM T55959 CI2VM7 11620991 Ki = 0.9 nM T55959 C5FQR2 11622909 Ki > 854 nM T55959 C1KD4Z 11623823 IC50 > 40000 nM T55959 C86SZO 11624458 IC50 = 21600 nM T55959 CYEH35 11627756 Ki = 6.9 nM T55959 C0I1YV 11628203 Ki = 2.2 nM T55959 CA8IM9 11630375 IC50 = 11 nM T55959 CF0QR8 11630988 Ki = 53 nM T55959 CXJ73O 11638552 Ki = 2200 nM T55959 CQ1U9W 11638962 Ki = 3670 nM T55959 C3VOG6 11644931 IC50 = 757 nM T55959 C97OLY 11649733 Ki = 0.4 nM T55959 CX2ZD7 11650267 Ki = 2478 nM T55959 C7BM5S 11650367 Ki = 6.3 nM T55959 C3OC6J 11650990 Ki = 27 nM T55959 C1HDM5 11653679 Ki = 1150 nM T55959 CL4AJ0 11658719 IC50 = 2532 nM T55959 CF92SM 11659664 Ki = 640 nM T55959 C0KH7D 11660186 IC50 = 10200 nM T55959 CIX54K 11666319 IC50 = 78 nM T55959 CJ9Z8D 11671232 Ki = 3.8 nM T55959 C98NXK 11671382 Ki = 1.6 nM T55959 CT3BP5 11674529 Ki = 3730 nM T55959 C79PHA 11678447 Ki = 0.8 nM T55959 C5Q3ZU 11680542 Ki = 79.43 nM T55959 C2DBG7 11687579 IC50 = 270 nM T55959 C0Y6OR 11687843 Ki = 2920 nM T55959 C8R7TP 11694495 IC50 = 509 nM T55959 C6T8ZD 11694789 IC50 = 110 nM T55959 CL19UR 11701869 IC50 = 4.5 nM T55959 CYN4H9 11702602 Ki > 200 nM T55959 C5OZD6 11706276 Ki = 1.8 nM T55959 CZB5P9 11709831 Ki = 3500 nM T55959 C4M9AU 11710505 Ki > 10000 nM T55959 CQWL60 11713341 Ki = 2.1 nM T55959 C18ZHK 11713731 Ki = 0.5 nM T55959 CHRM03 11716290 IC50 = 36350 nM T55959 CKQ03I 11716308 IC50 = 4589 nM T55959 CN2L4J 11716660 IC50 = 5.1 nM T55959 C9BD4J 11723014 Ki = 1210 nM T55959 C7PVL8 11730467 IC50 = 954 nM T55959 C4MC2V 11740717 Ki = 840 nM T55959 CD9E3Q 11748079 IC50 = 430 nM T55959 C2QZI5 11771101 Ki > 1000 nM T55959 CN4Y8B 11778700 IC50 = 373 nM T55959 CS54NA 11778793 IC50 = 47 nM T55959 CKNE31 11791987 Ki = 2800 nM T55959 CW15BI 11794260 Ki > 10000 nM T55959 C95EXO 11795979 Ki = 338.84 nM T55959 CQGL96 11797680 Ki = 0.45 nM T55959 CDH95C 11799242 Ki = 30.2 nM T55959 CA6GF2 11808524 IC50 = 113 nM T55959 CN9M8E 11811722 IC50 = 2250 nM T55959 CF2HI9 11812805 Ki = 48.98 nM T55959 CJO0Q6 11818515 Ki = 3549 nM T55959 C9ZQ4F 11826809 Ki = 16 nM T55959 C2UT9D 11846746 IC50 = 4430 nM T55959 CXLW54 11948707 Ki > 10000 nM T55959 C8EJ6H 11949672 IC50 > 10000 nM T55959 CK13QD 11953409 Ki = 6500 nM T55959 C8JQL7 11957735 IC50 > 10000 nM T55959 C0OF1U 11960210 IC50 = 1400 nM T55959 C5QB3M 11963972 IC50 = 2700 nM T55959 CAW2Y1 12000105 Ki = 756 nM T55959 C3LG9X 12017337 Ki = 48 nM T55959 CX2TQ7 12111555 IC50 = 246 nM T55959 C49HJG 12122109 Ki = 2000 nM T55959 CT4RA6 12204576 Ki = 1.7 nM T55959 CK6WG1 12276477 IC50 = 6043 nM T55959 C2MP5H 12559279 IC50 > 10000 nM T55959 CV70JI 12634880 Ki = 8 nM T55959 C6MH2K 12646716 IC50 = 543 nM T55959 C0KR1M 12884652 Ki = 450 nM T55959 CE5Y2W 12980713 IC50 = 1.43 nM T55959 CM78FI 12999584 IC50 = 3861 nM T55959 CCG14E 13091356 Ki = 620 nM T55959 CYN95Z 13091359 Ki = 1081 nM T55959 CU2Y5Z 13269476 Ki = 3600 nM T55959 CQV86I 13718739 IC50 > 10000 nM T55959 CGY6Q3 13718746 IC50 > 10000 nM T55959 C0KU4R 13718753 IC50 > 10000 nM T55959 C12NSL 13718761 IC50 > 10000 nM T55959 CI6TP9 13903189 Ki = 5.2 nM T55959 CHJ27K 13903191 Ki = 1.6 nM T55959 C4KU1J 14014888 IC50 > 10000 nM T55959 CQI9F6 14571114 Ki = 129 nM T55959 C9GEN5 14674210 IC50 = 670 nM T55959 CU08BA 14831998 IC50 = 33.7 nM T55959 C57QFI 14930273 Ki = 0.12 nM T55959 C7VAI1 15011772 IC50 > 10000 nM T55959 C0P5LY 15069893 IC50 = 6.5 nM T55959 CE4T7Z 15069894 Ki = 2.7 nM T55959 C8SXL1 15069905 IC50 = 1.7 nM T55959 CMI6C8 15113388 Ki = 82 nM T55959 C27ZJA 15113390 Ki = 173 nM T55959 CD24IR 15115364 IC50 = 1800 nM T55959 CTZ61G 15132121 IC50 = 36 nM T55959 C2T1UK 15290836 IC50 = 97 nM T55959 CO6P8K 15405849 Ki = 40.99 nM T55959 CMP83C 15550585 IC50 = 9.6 nM T55959 C53JMI 15639786 Ki = 4 nM T55959 C1FLJ0 15639787 Ki = 3.9 nM T55959 C4OT1S 15639792 IC50 = 22.7 nM T55959 CDW7C5 15679192 IC50 = 1.2 nM T55959 C6US3O 15711850 Ki = 1870 nM T55959 C5PO3N 15711869 Ki > 30000 nM T55959 CIGO41 15950719 IC50 = 3400 nM T55959 CW8M6S 15952123 IC50 = 2300 nM T55959 CM6O3G 15983286 IC50 = 813 nM T55959 C89XFJ 16007138 IC50 = 3.8 nM T55959 C7EX4C 16007262 IC50 = 5 nM T55959 C37FIP 16047544 Ki > 10000 nM T55959 C30UFT 16066811 IC50 = 3120 nM T55959 CH74RZ 16102752 IC50 = 32 nM T55959 C6OR3H 16102755 Ki = 3.6 nM T55959 C9SH0B 16102756 IC50 = 60 nM T55959 CA75KZ 16102757 Ki = 9.4 nM T55959 C1L9HQ 16102758 Ki = 130 nM T55959 CMUI02 16102759 IC50 = 370 nM T55959 CLO54U 16102760 Ki = 24 nM T55959 C3SEF2 16102761 IC50 = 290 nM T55959 CYF03S 16102762 IC50 = 240 nM T55959 C4N9BG 16102763 IC50 = 27 nM T55959 C2HLF8 16102765 Ki = 2.3 nM T55959 CTX94E 16102766 Ki = 1 nM T55959 C9HLB7 16102767 Ki = 52 nM T55959 CLHY18 16102768 Ki = 22 nM T55959 CG90ID 16102769 Ki = 3300 nM T55959 CH53XS 16102770 Ki = 6.6 nM T55959 CJ32XS 16113210 IC50 = 129 nM T55959 C9UYE0 16126667 Ki = 96 nM T55959 C4QCP3 16494915 IC50 > 10 nM T55959 C2VQS3 16640939 IC50 > 10000 nM T55959 C6P4BX 16656803 IC50 = 50 nM T55959 CZ2IS9 16660294 Ki > 2536 nM T55959 CW40DA 16678084 IC50 = 5329 nM T55959 CH4Y2D 16681434 IC50 = 9550 nM T55959 CDT5V8 16721129 Ki = 29 nM T55959 CL5G7A 16730754 Ki = 79 nM T55959 C50YME 16747877 Ki = 28 nM T55959 CY8QO6 16748004 Ki = 35 nM T55959 CY2FL4 16748005 Ki = 6.1 nM T55959 C9CQ1B 16748006 Ki = 8.6 nM T55959 COGJ31 16748007 Ki = 130 nM T55959 CPF2K0 16748165 Ki = 14 nM T55959 CM1L6Q 16748381 IC50 = 212 nM T55959 CG5FU0 16748382 Ki = 61 nM T55959 CYN9W8 16748383 Ki = 140 nM T55959 CM89SX 16748512 Ki = 53 nM T55959 C1ZQX9 16748513 Ki = 529 nM T55959 CM46NI 16748623 Ki = 7.7 nM T55959 C9W7LH 16748731 Ki = 12 nM T55959 CJ9S7I 16748848 Ki = 12 nM T55959 CXH10U 16748849 Ki = 39 nM T55959 C37DZJ 16748949 Ki = 66 nM T55959 CTJ2Z3 16748950 Ki = 212 nM T55959 C1L8DV 16748951 Ki = 105 nM T55959 CTI89R 16759249 Ki = 47 nM T55959 C7WHG3 17758197 Ki = 13.18 nM T55959 CN4HB8 18391094 IC50 = 12.6 nM T55959 CH39LP 18391096 IC50 = 690 nM T55959 CUEV14 18446803 IC50 = 19.4 nM T55959 C03IZO 18623856 Ki = 1.1 nM T55959 CJ6ZF2 18756309 IC50 = 546 nM T55959 C9JD5Y 19360456 IC50 = 300 nM T55959 CYFJ81 19926671 IC50 = 100 nM T55959 C21LXU 20055336 Ki = 290 nM T55959 C8ICF9 20111627 IC50 = 28 nM T55959 CQ6PB2 20443021 Ki = 4 nM T55959 CPVF37 20443023 Ki = 6.5 nM T55959 CX9HZ2 20443040 Ki = 54 nM T55959 CC2G4J 20611340 IC50 = 0.57 nM T55959 C6R8AM 20631904 Ki = 43 nM T55959 C81FRQ 20636465 Ki = 31 nM T55959 CXQM78 20695745 IC50 = 2060 nM T55959 CEO8W1 21116177 IC50 = 437 nM T55959 C5RNG7 21121582 Ki = 14.13 nM T55959 CRV56X 21365270 IC50 = 26 nM T55959 C3T5HF 21509921 Ki > 10000 nM T55959 CFN81Q 21527771 Ki > 10000 nM T55959 CH59WN 21533446 Ki = 497 nM T55959 C9H4XW 21539375 IC50 = 81.5 nM T55959 C27GSH 21539381 IC50 = 179.3 nM T55959 C1MR4F 21959106 IC50 = 0.49 nM T55959 C42AIN 21959117 IC50 = 408 nM T55959 C0AW7O 21959124 IC50 = 0.66 nM T55959 C2X0TW 22337167 IC50 > 100000 nM T55959 CR4T9J 22337182 Ki > 100000 nM T55959 CQUY92 22386812 Ki = 107 nM T55959 C7O8WZ 22386894 Ki = 10.9 nM T55959 CMDI47 22386922 Ki = 157 nM T55959 CW5M2S 22419110 IC50 = 27.8 nM T55959 C51XVN 22419115 IC50 = 1100 nM T55959 CPI8Q3 22419116 IC50 = 7.93 nM T55959 CU8YV6 22468266 Ki = 25 nM T55959 CF6P4V 22468271 Ki = 430 nM T55959 CV2XH0 22798952 IC50 = 1584.89 nM T55959 CD63RO 22860156 IC50 = 3380 nM T55959 C1KT4Z 22896736 Ki = 16 nM T55959 CL97PH 22896763 Ki = 9.7 nM T55959 CPH6L4 22966050 Ki = 2240 nM T55959 CYPV48 23378645 IC50 = 640 nM T55959 C4ATJ7 23378652 IC50 = 1800 nM T55959 C57EFO 23378743 IC50 = 5800 nM T55959 C2QXK6 23449967 IC50 = 68 nM T55959 CUD3Y7 23449968 IC50 = 2.34 nM T55959 CMEV08 23449969 IC50 = 1900 nM T55959 CCP24F 23449972 IC50 = 390 nM T55959 C31ASG 23449975 IC50 = 22 nM T55959 C2HK1Z 23449980 IC50 = 7 nM T55959 CP1A4B 23449981 IC50 = 62 nM T55959 CW0D5K 23449986 IC50 = 28.5 nM T55959 CH8O4R 23449987 IC50 = 3816 nM T55959 CG08BF 23449988 IC50 = 238 nM T55959 CHD8T7 23449989 IC50 = 2730 nM T55959 C7YFT3 23582127 Ki = 983 nM T55959 C57MTL 23625757 Ki = 190 nM T55959 CK1A0B 23661668 Ki = 67900 nM T55959 C6IF2N 23661687 Ki = 60 nM T55959 CSB9E8 24103136 IC50 = 5400 nM T55959 C0I5RA 24180665 IC50 = 260 nM T55959 C91IVZ 24742317 IC50 > 10000 nM T55959 C32IVO 24742475 IC50 = 5100 nM T55959 CWGH86 24743352 IC50 = 5539 nM T55959 CYBG40 24743354 IC50 > 10000 nM T55959 CG3XD5 24743436 IC50 = 3600 nM T55959 C61QPT 24748794 Ki = 351 nM T55959 C9P2NE 24748795 Ki = 443 nM T55959 CYRZ48 24749837 Ki > 1000 nM T55959 C4Y0BF 24749952 Ki > 1000 nM T55959 CJ2N8B 24749953 Ki = 576 nM T55959 CV30EH 24749955 Ki > 1000 nM T55959 CPD4M8 24749956 Ki > 1000 nM T55959 CO7TD4 24750311 Ki = 340 nM T55959 C4R9YO 24750312 Ki = 847 nM T55959 C60SIH 24750313 Ki > 1000 nM T55959 C2ZJ3Q 24750421 Ki = 299 nM T55959 CV1K6O 24750422 Ki > 1000 nM T55959 CQ1G3S 24750423 Ki = 659 nM T55959 CHI83W 24769038 IC50 = 2.8 nM T55959 C5ASY1 24773552 Ki = 221 nM T55959 C1FIS5 24773804 Ki > 2000 nM T55959 C9KXC8 24773805 Ki > 2000 nM T55959 CP1F6M 24782241 Ki = 6.31 nM T55959 CZ2XE7 24782243 Ki = 3.162 nM T55959 CJQ2X4 24782485 Ki = 15.85 nM T55959 CI7S2G 24782486 Ki = 15.85 nM T55959 CK5TO1 24782487 Ki = 501.19 nM T55959 CZ34RN 24782489 Ki = 79.43 nM T55959 CL5GS1 24786064 Ki = 125.89 nM T55959 CQN4W1 24802843 Ki = 79.43 nM T55959 C23ICW 24802846 Ki = 25.12 nM T55959 CX6ZB7 24802848 Ki = 31.62 nM T55959 CH30VR 24803009 Ki = 251.19 nM T55959 CH87VD 24803010 Ki = 3.981 nM T55959 CC78ZE 24803012 Ki = 39.81 nM T55959 C7C4UQ 24803014 Ki = 3162.28 nM T55959 C17ISZ 24803180 Ki = 7943.28 nM T55959 C4O8ZF 24803181 Ki = 1584.89 nM T55959 C1W8NS 24803185 Ki = 158.49 nM T55959 C9LV3D 24803344 Ki = 39.81 nM T55959 C96CBA 24803345 Ki = 398.11 nM T55959 CPH72B 24825320 Ki = 39 nM T55959 C3LW5Z 24825321 Ki = 20 nM T55959 CHZS54 24825322 Ki = 29 nM T55959 C03LDP 24825323 Ki = 27 nM T55959 C2IB8H 24825324 Ki = 2.7 nM T55959 CQKH10 24825325 Ki = 22 nM T55959 CPN0C7 24825326 Ki = 18 nM T55959 CAV1B6 24825327 Ki = 30 nM T55959 C0BR5C 24825328 Ki = 7 nM T55959 CVQ8C7 24825329 Ki = 10 nM T55959 CV72IA 24825330 Ki = 100 nM T55959 CL0DF1 24825331 Ki = 410 nM T55959 CR2L5Q 24825332 Ki = 57 nM T55959 C9V6HW 24825333 Ki = 150 nM T55959 CAD2R1 24825334 Ki = 450 nM T55959 CR3FA2 24825335 Ki = 140 nM T55959 C17ZME 24825336 Ki = 110 nM T55959 C0M7CN 24825720 Ki = 478.63 nM T55959 CDC91N 24839550 Ki = 1258.93 nM T55959 CY21RE 24841480 Ki = 970 nM T55959 C6ZRA7 24849533 Ki = 63.1 nM T55959 C50XIV 24855884 Ki = 330 nM T55959 CJTY89 24855886 Ki = 9000 nM T55959 C79FCO 24855918 Ki = 8000 nM T55959 CJAC42 24855949 Ki = 7300 nM T55959 C1SVD5 24855952 Ki = 7700 nM T55959 C0DUL3 24857666 IC50 = 350 nM T55959 CC8J1Z 24857667 IC50 = 408 nM T55959 C9V5MT 24857668 IC50 = 894 nM T55959 C5QGY4 24857669 IC50 = 175 nM T55959 CSR8J4 24857759 IC50 = 32 nM T55959 C27EUV 24857839 IC50 > 10000 nM T55959 CZ8TA6 24857854 IC50 > 10000 nM T55959 C97SEP 24857858 Ki = 2490 nM T55959 CBI5D7 24860769 IC50 = 2300 nM T55959 C7COU6 24860831 IC50 = 29 nM T55959 CVO64M 24860832 IC50 = 4000 nM T55959 CL26KS 24860835 IC50 = 120 nM T55959 C7EHG5 24860898 IC50 = 996 nM T55959 C2X6VF 24860899 IC50 = 530 nM T55959 CAU07P 24860900 IC50 = 1000 nM T55959 CM9L7D 24860902 IC50 = 75 nM T55959 CZ3R7W 24860903 IC50 < 1 nM T55959 CG8T3J 24860904 IC50 = 180 nM T55959 CO51AG 24863961 Ki = 6331 nM T55959 CD9SF2 24863962 Ki = 4123 nM T55959 CXD45U 24867041 IC50 = 96 nM T55959 CV1PY2 24878951 Ki = 2389 nM T55959 CK6JC4 24878953 Ki = 13190 nM T55959 C4SL0V 24879001 Ki = 9530 nM T55959 C3Z4JN 24879003 Ki > 10000 nM T55959 C56IDA 24879005 Ki = 5525 nM T55959 C23LNY 24879008 Ki = 11970 nM T55959 C9C8OH 24879010 Ki = 11920 nM T55959 C1ZRH6 24879054 Ki > 10000 nM T55959 CD17RE 24879056 Ki > 10000 nM T55959 CX20BZ 24879058 Ki > 10000 nM T55959 C9A2NF 24890939 Ki = 490 nM T55959 CG0Z8X 24893996 IC50 = 5800 nM T55959 CYKD83 24894907 Ki = 235 nM T55959 C0EYS5 24895131 Ki = 73 nM T55959 C4FEQ6 24936132 Ki > 9000 nM T55959 CF2A7C 24936614 IC50 = 512 nM T55959 C3H5PJ 24947569 Ki = 8300 nM T55959 C4Y7FP 24947750 Ki = 7300 nM T55959 CA8VN2 24947751 Ki = 4000 nM T55959 CYGT57 24947752 Ki = 7000 nM T55959 CEW8C3 24947936 Ki = 7000 nM T55959 C6BIR1 24947941 Ki = 7000 nM T55959 C06TLI 24948121 Ki = 3000 nM T55959 CW4X0E 24962988 Ki = 3030 nM T55959 CQ42YZ 24964158 Ki = 700 nM T55959 C4P5AD 24964159 Ki = 1000 nM T55959 CB9C4E 24965063 Ki > 6000 nM T55959 CZXC58 24965064 Ki > 6000 nM T55959 CT39VO 24969452 IC50 = 10000 nM T55959 CGZ60N 24969453 IC50 = 8000 nM T55959 CZ6T5Q 25009937 Ki = 1570 nM T55959 CQ9LS6 25022704 Ki = 1910 nM T55959 C0HRL1 25024305 Ki = 7.943 nM T55959 C2RQX9 25024309 Ki = 10 nM T55959 C3W1NC 25024503 Ki = 251.19 nM T55959 CY0VU5 25025577 Ki = 512.86 nM T55959 CA20NZ 25025581 IC50 = 5.012 nM T55959 CU8A6N 25025776 Ki = 12.59 nM T55959 C4I5LJ 25025778 Ki = 25.12 nM T55959 CPJD86 25025779 Ki = 25.12 nM T55959 CN0U3C 25025780 Ki = 39.81 nM T55959 CFAZ02 25025782 Ki = 7.943 nM T55959 CDX2C6 25025977 Ki = 5.012 nM T55959 CRQ73B 25025978 Ki = 12.59 nM T55959 C9WQ5K 25025979 Ki = 2.512 nM T55959 CA4L5Q 25032786 IC50 > 10 nM T55959 C6K4SH 25033519 IC50 = 195 nM T55959 CPT9X8 25066443 IC50 = 5040 nM T55959 CIWT97 25071015 Ki = 343 nM T55959 CP9J7Q 25071019 IC50 > 10000 nM T55959 C0YEI8 25141192 IC50 = 1.57 nM T55959 C0MPE3 25141372 Ki > 1000 nM T55959 C0OT1F 25141373 Ki > 1500 nM T55959 C7W9YX 25150535 IC50 > 10000 nM T55959 C35XQI 25150621 IC50 > 10000 nM T55959 CD0QU5 25150624 IC50 > 10000 nM T55959 CIZ1N9 25150625 IC50 > 10000 nM T55959 C6IXV9 25150627 IC50 > 10000 nM T55959 CE1ND3 25150628 IC50 > 10000 nM T55959 CAVR45 25150711 IC50 > 10000 nM T55959 CW9MX8 25168440 Ki = 18 nM T55959 CXC35U 25168857 IC50 > 10000 nM T55959 CZ86GS 25181041 Ki = 275.42 nM T55959 C7JYI8 25188212 Ki > 6000 nM T55959 C56CDP 25188770 Ki = 327 nM T55959 C5Z0LT 25188771 Ki > 6000 nM T55959 C46ANM 25195291 Ki = 3190 nM T55959 C37YTG 25210603 Ki = 6.31 nM T55959 CW3JR1 25210604 Ki = 25.12 nM T55959 CCTO39 25210872 Ki = 7.943 nM T55959 CE7BA0 25210873 Ki = 10 nM T55959 C0FE8U 25210874 Ki = 15.85 nM T55959 C0XN3L 25210876 Ki = 6.31 nM T55959 CF6AD3 25211583 Ki = 2716 nM T55959 CVU7J1 25211682 Ki = 4492 nM T55959 CJ1Z9H 25216680 Ki > 10000 nM T55959 C1T3LR 25218143 Ki > 10000 nM T55959 CPI03N 25218397 Ki > 10000 nM T55959 CL1R3Q 25218401 Ki > 10000 nM T55959 CX07CK 25258806 IC50 > 100000 nM T55959 CHY8S9 25258809 Ki = 66988 nM T55959 CNR21Q 25260901 Ki = 290 nM T55959 C7PK2X 29938807 Ki = 9.3 nM T55959 CSO5Y3 29981497 Ki = 130000 nM T55959 CN8J0W 29981513 Ki = 3509000 nM T55959 CJ1N0X 29981679 Ki = 2814000 nM T55959 CH3M1E 31413243 IC50 > 10000 nM T55959 C9GS1N 31413320 IC50 > 10000 nM T55959 C2XY4V 31413484 IC50 > 10000 nM T55959 C4FR6G 36465568 IC50 > 10000 nM T55959 C1J4XZ 42636222 IC50 = 2113 nM T55959 CR70ZY 43164282 IC50 = 150 nM T55959 CNL52R 43283283 IC50 = 506 nM T55959 C6P5DK 43283415 IC50 = 421 nM T55959 C1YM3D 44131466 Ki = 6410 nM T55959 CMTB93 44131470 Ki = 2590 nM T55959 CYE20L 44131666 Ki > 6320 nM T55959 CPR7L3 44133672 Ki = 6650 nM T55959 CE3SD9 44133859 Ki = 310 nM T55959 CZ2VQ1 44133861 Ki > 5500 nM T55959 C9P5XU 44133863 Ki > 6140 nM T55959 C2G7AO 44134036 Ki > 6370 nM T55959 C5YKI9 44134038 Ki > 6180 nM T55959 C6DQJ3 44134039 Ki > 6630 nM T55959 C8RZX0 44134041 Ki > 6650 nM T55959 CW5Q9P 44143473 Ki = 7307 nM T55959 CFP9S1 44157038 Ki > 10000 nM T55959 CO0GC4 44157259 Ki > 6000 nM T55959 CGA8B4 44157339 Ki > 6000 nM T55959 C25DHI 44178203 Ki = 158.49 nM T55959 CI12UH 44188274 IC50 > 40000 nM T55959 CT30BL 44188275 IC50 > 30000 nM T55959 CH7FJ6 44188689 Ki = 63.1 nM T55959 CSE8X3 44188690 Ki = 794.33 nM T55959 CY2Q9O 44188691 Ki = 25.12 nM T55959 C6FPM5 44188693 Ki = 31.62 nM T55959 CWR04I 44188695 Ki = 15.85 nM T55959 CJEG24 44188861 Ki = 199.53 nM T55959 C9XSI6 44189029 Ki = 316.23 nM T55959 C2AV1K 44190762 IC50 = 3410 nM T55959 C6WSI1 44204599 IC50 = 1.93 nM T55959 C2KJB0 44216880 Ki = 83 nM T55959 CA50PK 44219207 Ki = 6.31 nM T55959 CQY1J3 44219363 Ki = 25.12 nM T55959 CJX5T2 44219364 Ki = 25.12 nM T55959 C6SF0L 44219365 Ki = 1.995 nM T55959 CWP84D 44219367 Ki = 125.89 nM T55959 CVG5I0 44219517 Ki = 19.95 nM T55959 C1NQ2R 44219519 Ki = 12.59 nM T55959 CKMV39 44219520 Ki = 12.59 nM T55959 CA46YO 44230734 Ki = 39 nM T55959 CCK73R 44230855 IC50 = 470 nM T55959 CB5P7N 44230873 Ki = 62 nM T55959 CXI7Z8 44230875 Ki = 58 nM T55959 CU8MS7 44230877 Ki = 724 nM T55959 C67PRE 44231009 Ki = 21 nM T55959 C67WIP 44231010 Ki = 550 nM T55959 CCP13S 44231144 Ki = 115 nM T55959 CIBR82 44231149 Ki = 331 nM T55959 CE12BT 44231265 Ki = 104 nM T55959 C0TF4H 44231266 Ki = 38 nM T55959 C7HCZ5 44231267 Ki = 363 nM T55959 CDZ8F4 44231268 Ki = 741 nM T55959 C0AW6X 44241240 IC50 = 190 nM T55959 C8AFN4 44241291 IC50 = 340 nM T55959 C63GVH 44241292 IC50 = 130 nM T55959 CZXC86 44267871 Ki = 81 nM T55959 C8WZG7 44269522 Ki = 3.1 nM T55959 C0MCK3 44269548 Ki = 6.73 nM T55959 C96ZRI 44269549 Ki = 22 nM T55959 C5YE8A 44269598 Ki = 5.6 nM T55959 CI14GD 44269607 Ki = 3.9 nM T55959 CE20CZ 44275807 Ki = 4897.79 nM T55959 CO52EQ 44276147 IC50 = 377 nM T55959 CZ30EN 44276148 IC50 = 166 nM T55959 C1DMB7 44276228 IC50 = 3.5 nM T55959 C1UDT3 44290461 IC50 = 1.4 nM T55959 C1QHI4 44295709 IC50 = 1.08 nM T55959 C2B8AN 44295896 IC50 = 0.6 nM T55959 CC3T9P 44295975 IC50 = 1.7 nM T55959 C8DKL9 44296390 Ki = 1.8 nM T55959 CEO46F 44305466 Ki = 910 nM T55959 C97SYT 44305491 Ki = 3320 nM T55959 CZG6F3 44305492 Ki = 3600 nM T55959 CD3M2K 44307360 Ki = 8.83 nM T55959 CUSR03 44307440 Ki = 438 nM T55959 C3WLT2 44307441 Ki = 29.8 nM T55959 C7U8NC 44307585 Ki = 54 nM T55959 C8RHD9 44308474 Ki = 18.4 nM T55959 C0LCV4 44308475 Ki = 21.7 nM T55959 C0O2BH 44308682 IC50 = 52.2 nM T55959 C38IFX 44321638 IC50 = 123 nM T55959 CX1EB8 44322005 IC50 = 7.7 nM T55959 C1B4LU 44322022 IC50 = 6300 nM T55959 CV7NH3 44322023 IC50 = 1.1 nM T55959 C7S2VP 44322076 IC50 = 235 nM T55959 CI0GO4 44322143 IC50 = 55.1 nM T55959 CQHJ59 44322164 IC50 = 3530 nM T55959 CI90PQ 44322194 IC50 > 20000 nM T55959 CBN85G 44322218 IC50 = 2590 nM T55959 CGA75L 44322219 IC50 = 7730 nM T55959 CV1Q8O 44322257 IC50 = 2.8 nM T55959 CLY2O1 44322269 IC50 = 477 nM T55959 CH0T6J 44322276 IC50 = 3.02 nM T55959 C9APJ1 44322284 IC50 = 45 nM T55959 CP21ST 44322286 IC50 = 448 nM T55959 C5DVG7 44322287 IC50 = 3.04 nM T55959 CU7R1K 44322314 IC50 = 1.19 nM T55959 CB4V5Y 44322477 IC50 = 33.2 nM T55959 CNMH73 44322592 IC50 = 0.3 nM T55959 CG5L9Y 44322645 IC50 > 10000 nM T55959 C0PXM6 44322646 IC50 > 150000 nM T55959 C1WFT6 44323041 IC50 = 3840 nM T55959 CJQ5A4 44323053 IC50 = 21900 nM T55959 CZ0W9D 44323131 IC50 = 22300 nM T55959 C5JKV9 44323133 IC50 = 20300 nM T55959 CE1T8P 44323347 IC50 = 10.9 nM T55959 CM8GB2 44323348 IC50 > 10000 nM T55959 CFG7W3 44323488 IC50 = 520 nM T55959 C5VN6Y 44332279 IC50 = 787 nM T55959 C16GET 44332309 IC50 = 335 nM T55959 CU0SQ8 44332340 IC50 = 3320 nM T55959 C1E9NU 44332360 IC50 = 11 nM T55959 C2MFB8 44332404 IC50 = 42 nM T55959 C6F4XC 44332405 IC50 = 25 nM T55959 C78AWT 44332801 IC50 = 390 nM T55959 CK68BR 44332802 IC50 = 570 nM T55959 CEG5D6 44332819 IC50 = 538 nM T55959 CICR35 44340153 Ki = 60 nM T55959 CJL61A 44340169 Ki = 41 nM T55959 C40RKF 44340181 Ki = 25 nM T55959 C78CFJ 44340203 Ki = 38 nM T55959 CB34ZC 44340445 Ki = 64 nM T55959 CVWM21 44340483 Ki = 50 nM T55959 C4TSF5 44340484 Ki = 6 nM T55959 CQL94N 44340485 Ki = 72 nM T55959 C1OD0T 44341910 Ki = 48.98 nM T55959 CWS89Y 44341929 Ki = 14.13 nM T55959 C1PF3E 44341939 Ki = 8.128 nM T55959 CN56QP 44341940 Ki = 22.39 nM T55959 CRK2U0 44342076 Ki = 18.62 nM T55959 CAL61E 44342079 Ki = 229.09 nM T55959 C35RLE 44342204 Ki = 6.457 nM T55959 C0P9AW 44342206 Ki = 660.69 nM T55959 C51NOI 44344091 Ki > 10000000 nM T55959 CX12US 44344115 Ki = 7275000 nM T55959 C4PT6K 44344218 Ki = 353000 nM T55959 CX2O9B 44344235 Ki = 240500 nM T55959 CZ4S1N 44346228 IC50 = 490 nM T55959 C4QXL7 44346323 Ki = 4140 nM T55959 CEV3J8 44346324 Ki = 8190 nM T55959 C30HGO 44346337 Ki = 3650 nM T55959 CM24FU 44346354 Ki = 10650 nM T55959 C1F0AZ 44346379 Ki = 4350 nM T55959 C47SLT 44348860 IC50 = 6030 nM T55959 C1A2DC 44348878 IC50 = 55.9 nM T55959 CQ54ET 44348881 IC50 = 1480 nM T55959 C5B8PU 44348886 IC50 = 389 nM T55959 CZU4K0 44348893 IC50 = 33.5 nM T55959 CQ7FV5 44348898 IC50 = 80.2 nM T55959 C1UQ8B 44348903 IC50 = 72 nM T55959 C97XUW 44348914 IC50 = 99 nM T55959 CD5I2E 44348915 IC50 = 119 nM T55959 C7PFJ2 44348927 IC50 = 22 nM T55959 C5YD7O 44348929 IC50 = 20.3 nM T55959 CV8GJ6 44348934 IC50 = 240 nM T55959 CFQ6K0 44348935 IC50 = 13.2 nM T55959 C95ESH 44348942 IC50 = 223 nM T55959 CX78DN 44348951 IC50 = 15.8 nM T55959 CV9LR5 44348952 IC50 = 49.5 nM T55959 CS3UM7 44349165 IC50 = 909 nM T55959 CU9VM1 44349166 IC50 = 91.4 nM T55959 C91DNF 44349181 IC50 = 24 nM T55959 CS56AC 44353682 IC50 = 36.1 nM T55959 CCI5T8 44354020 Ki > 10000 nM T55959 CGQ13N 44354021 Ki > 10000 nM T55959 C68QVH 44354105 IC50 = 507 nM T55959 C2TGL8 44354122 Ki > 10000 nM T55959 C4GVC5 44354236 Ki = 1536 nM T55959 CFW7N2 44358674 IC50 = 20.3 nM T55959 CUN25S 44358675 IC50 = 5.69 nM T55959 CJ36NW 44364204 Ki = 53 nM T55959 C0O2NU 44364206 Ki = 63 nM T55959 CMA5D4 44364314 Ki = 80 nM T55959 C69BCI 44364358 Ki = 280 nM T55959 CL2M6Y 44364359 Ki = 140 nM T55959 C35MGZ 44364439 Ki = 1100 nM T55959 CLW8D9 44364455 Ki = 8.1 nM T55959 CRY94A 44370219 Ki > 10000 nM T55959 CTB3Q6 44372823 Ki = 0.48 nM T55959 C5DA8L 44372825 Ki = 0.9 nM T55959 CWGQ58 44383909 Ki = 3.47 nM T55959 CP4JB9 44384015 IC50 = 28 nM T55959 CU8Z1R 44384016 IC50 = 32 nM T55959 C24DSJ 44384117 Ki = 1.88 nM T55959 C1BXI7 44395690 IC50 = 20 nM T55959 CEY74D 44395805 IC50 = 220 nM T55959 CZWE51 44395806 IC50 = 13 nM T55959 C7ZGQ3 44395831 IC50 = 910 nM T55959 CY2WM9 44395924 IC50 = 8 nM T55959 C0FV1Y 44395952 Ki = 5 nM T55959 C3C9VY 44395953 Ki = 5 nM T55959 CK5VX8 44396000 Ki = 5 nM T55959 CR29YA 44396039 Ki = 5 nM T55959 CG8WJ1 44396040 Ki = 5 nM T55959 CX0V4W 44398372 Ki > 1000 nM T55959 CA09EW 44404169 Ki > 200 nM T55959 C5Y8LB 44404175 Ki > 200 nM T55959 CM46ID 44404176 Ki > 200 nM T55959 CX02GP 44404182 Ki > 200 nM T55959 CV39CT 44404223 Ki > 200 nM T55959 C3KE9P 44404224 Ki > 200 nM T55959 CWD08P 44404228 Ki > 200 nM T55959 CG4P9S 44404235 Ki > 200 nM T55959 CVW0P1 44404239 Ki > 200 nM T55959 CZ9GU0 44404250 Ki > 200 nM T55959 CF8Z6A 44404254 Ki > 200 nM T55959 CN15FZ 44404255 Ki > 200 nM T55959 C30QXS 44404259 Ki > 200 nM T55959 C8U9NH 44404261 Ki > 200 nM T55959 CRSC86 44404262 Ki > 200 nM T55959 CM7W1J 44404265 Ki > 200 nM T55959 CFP8D2 44404266 Ki > 200 nM T55959 C97CAH 44404269 Ki = 13 nM T55959 C5R7XB 44404273 Ki > 200 nM T55959 C5F2VA 44404274 Ki > 200 nM T55959 CGN87C 44404278 Ki > 200 nM T55959 CSO98W 44404279 Ki > 200 nM T55959 CRIG21 44404285 Ki > 200 nM T55959 CO57NJ 44404286 Ki > 200 nM T55959 CL6C2S 44404914 IC50 = 28 nM T55959 CSDN32 44405146 Ki = 436 nM T55959 C4DFS7 44405156 Ki = 50 nM T55959 C56TNY 44405790 Ki = 24 nM T55959 CZI0A4 44405840 IC50 = 0.002 nM T55959 CR30FO 44405845 IC50 = 9350 nM T55959 C9TUH6 44405846 IC50 = 9240 nM T55959 CFT43Y 44405871 IC50 = 67000 nM T55959 CS2Q0A 44405875 IC50 = 7220 nM T55959 CR06US 44405876 IC50 = 603 nM T55959 CG3WT6 44405893 IC50 = 16800 nM T55959 CDF9N4 44405897 IC50 = 3980 nM T55959 C4GN3T 44405898 IC50 = 21900 nM T55959 CA3I0W 44407714 Ki = 3850 nM T55959 CIH46L 44408412 IC50 > 100 nM T55959 CK6O7A 44408415 IC50 > 100 nM T55959 CV3QD5 44408434 IC50 > 100 nM T55959 C7T6WF 44408435 IC50 > 100 nM T55959 CJ3NS2 44408441 IC50 > 100 nM T55959 CT52PU 44408442 IC50 > 100 nM T55959 CDQ34O 44408477 IC50 > 100 nM T55959 CI3Z8X 44408529 IC50 > 100 nM T55959 CYP8A5 44408580 IC50 > 100 nM T55959 CA3P6K 44408581 IC50 > 100 nM T55959 C6F5EC 44408582 IC50 > 100 nM T55959 CKX2P8 44408664 IC50 = 220 nM T55959 C3C9PW 44408718 IC50 = 100 nM T55959 CK9U7V 44408719 IC50 = 830 nM T55959 C83DCF 44408748 IC50 = 2500 nM T55959 CQ64UC 44408749 IC50 = 1100 nM T55959 C14BYG 44408753 IC50 = 29 nM T55959 CI0JZ2 44408756 IC50 = 55 nM T55959 C9U3TR 44408757 IC50 = 90 nM T55959 C6LTD5 44408760 IC50 = 250 nM T55959 CYAC79 44408761 IC50 = 360 nM T55959 CX2S0E 44408762 IC50 = 20 nM T55959 C3QCP2 44408802 IC50 = 1400 nM T55959 CLJ3U7 44408856 IC50 = 1300 nM T55959 C5K8NB 44408857 IC50 = 3300 nM T55959 C2QMD8 44408858 IC50 = 920 nM T55959 CI3ZS8 44408859 IC50 = 16700 nM T55959 C1ZPY7 44408870 IC50 = 290 nM T55959 C8ZH4C 44408871 IC50 = 420 nM T55959 C2J1KW 44408875 IC50 = 90 nM T55959 CZ8G2B 44408876 IC50 = 120 nM T55959 CKR78J 44408885 IC50 = 3600 nM T55959 CC9D8S 44408886 IC50 = 12900 nM T55959 CW7VA3 44408917 IC50 = 240 nM T55959 CBS73M 44408918 IC50 = 540 nM T55959 CQ45GH 44408921 IC50 = 5100 nM T55959 CKM7O2 44408922 IC50 = 89 nM T55959 C13IEG 44408925 IC50 = 375 nM T55959 CE5AC6 44408926 IC50 = 90 nM T55959 C2D5WU 44408969 IC50 < 1 nM T55959 CG87PW 44409290 Ki > 1000 nM T55959 C24AHO 44411099 Ki = 201 nM T55959 C2EQ1I 44411140 Ki = 240 nM T55959 CCBK16 44411148 Ki = 98 nM T55959 CQA1W4 44411179 Ki = 86.5 nM T55959 C60ECT 44411185 Ki = 200 nM T55959 C1VHP7 44411215 Ki = 330 nM T55959 C3M7RB 44411224 Ki = 230 nM T55959 CT7D0B 44411228 Ki = 190 nM T55959 CE5A4F 44411296 Ki = 160 nM T55959 C8GD7M 44411395 Ki = 83 nM T55959 C5ZN4X 44411491 Ki = 580 nM T55959 C6CW9U 44411501 Ki = 120 nM T55959 CIBG87 44413825 IC50 = 410 nM T55959 CFN48L 44413826 IC50 = 130 nM T55959 CA97VC 44413836 IC50 = 390 nM T55959 CLG5H8 44413837 IC50 > 2000 nM T55959 CCY43Q 44413856 IC50 = 160 nM T55959 CW0VE9 44413857 IC50 = 170 nM T55959 C05UKL 44413866 IC50 = 290 nM T55959 CCJ4X1 44413903 IC50 = 1920 nM T55959 C81IAE 44413904 IC50 = 150 nM T55959 C5Z2GC 44413925 IC50 = 490 nM T55959 C3BMI9 44413953 IC50 = 890 nM T55959 C18JHP 44413959 IC50 = 70 nM T55959 CNR87Z 44414690 IC50 = 2300 nM T55959 CM9V8F 44414692 IC50 = 1600 nM T55959 CQD2S5 44414696 Ki > 10000 nM T55959 CZ9LM3 44414707 IC50 > 4000 nM T55959 C9XIR1 44414734 IC50 > 4000 nM T55959 C81QHB 44414760 IC50 > 4000 nM T55959 CV37KC 44414761 IC50 > 4000 nM T55959 C3LJ7N 44414780 IC50 = 970 nM T55959 CY5Q9A 44414800 IC50 = 9200 nM T55959 C3RZ0N 44414809 IC50 > 4000 nM T55959 CF8Q6Y 44414836 IC50 > 4000 nM T55959 CJ8C0P 44415527 IC50 = 11 nM T55959 C4C9LS 44415528 IC50 = 36 nM T55959 CVTQ68 44416033 Ki = 41.92 nM T55959 CZ6WJ8 44416034 Ki = 12.25 nM T55959 CRA8M1 44416084 Ki = 8.48 nM T55959 C1BF0K 44416103 Ki = 13.25 nM T55959 C9Q5UZ 44416104 Ki = 2.94 nM T55959 C9UDS3 44416105 Ki = 4.54 nM T55959 CHF6L7 44417598 Ki = 29.9 nM T55959 CK5PZ8 44417599 Ki = 32.6 nM T55959 CRZK78 44418862 Ki = 1.4 nM T55959 CXA51W 44419295 Ki = 451 nM T55959 CLA67J 44419296 Ki = 609 nM T55959 C82VQX 44419298 Ki = 754 nM T55959 CRAK93 44419299 Ki = 2659 nM T55959 CZT81O 44419300 Ki = 651 nM T55959 C2WDJ5 44419301 Ki = 621 nM T55959 C85OTF 44419303 Ki = 931 nM T55959 CZ5O8Y 44419306 Ki = 1224 nM T55959 CXP1A6 44419308 Ki = 2082 nM T55959 CM3K1F 44419314 Ki = 10 nM T55959 CG8F3J 44419327 Ki = 32 nM T55959 CJR7P1 44419328 Ki = 219 nM T55959 C7DQL6 44419331 Ki = 119 nM T55959 CVMF25 44419335 Ki = 251 nM T55959 C59ZPV 44419340 Ki = 855 nM T55959 C71CPW 44419344 Ki = 157 nM T55959 CM1WZ9 44419345 Ki = 297 nM T55959 CJHN07 44421413 IC50 = 101 nM T55959 CEHO31 44421414 IC50 = 21 nM T55959 C2WE3K 44421423 IC50 = 1.7 nM T55959 C1S3RH 44421438 IC50 = 11.7 nM T55959 CSIN57 44421439 IC50 = 23.4 nM T55959 CQI4V3 44421455 IC50 = 10.2 nM T55959 C2BEZ9 44421482 IC50 = 340 nM T55959 C7PCA5 44421483 IC50 = 1.23 nM T55959 CNYK42 44421484 IC50 = 23.3 nM T55959 CB17LT 44421485 IC50 = 980 nM T55959 CE6G3H 44421486 IC50 = 0.9 nM T55959 CL6M9V 44421497 IC50 = 1.96 nM T55959 CSU23Q 44421500 IC50 = 22.4 nM T55959 CL1V7W 44422784 IC50 = 2 nM T55959 CV43NH 44427225 IC50 = 2000 nM T55959 CGX49R 44427889 Ki = 13 nM T55959 C7I2MZ 44427901 Ki = 13 nM T55959 CGOD89 44429174 Ki = 322 nM T55959 C6BW5V 44429184 Ki = 1250 nM T55959 CIJ5R2 44429185 Ki = 922 nM T55959 C6OVA2 44429187 Ki = 20600 nM T55959 CNP37Y 44429189 Ki = 1900 nM T55959 C8SR0G 44429190 Ki = 2100 nM T55959 C53AFL 44429191 Ki = 3300 nM T55959 CN4UT8 44429192 Ki = 4100 nM T55959 C5HK8Y 44429193 Ki = 6300 nM T55959 C7J6GA 44429194 Ki = 302000 nM T55959 CK9H1C 44429195 Ki = 2649000 nM T55959 CQA0W7 44429197 Ki = 49000 nM T55959 CV9M4N 44429198 Ki = 121000 nM T55959 CUH0B6 44429199 Ki = 6540 nM T55959 CS2ER7 44429200 Ki = 625 nM T55959 CE2M3T 44429201 Ki = 589 nM T55959 CE31CZ 44429202 Ki = 22000 nM T55959 CF5CO6 44429203 Ki = 1500 nM T55959 CJ9VZ1 44429204 Ki = 264000 nM T55959 CJ5F4X 44429205 Ki = 605000 nM T55959 CLK84J 44429206 Ki = 1660000 nM T55959 CH50DU 44429207 Ki = 630000 nM T55959 C1Z7KB 44429209 Ki = 1050000 nM T55959 C7OQT6 44429210 Ki = 590000 nM T55959 CI46CX 44429212 Ki = 231000 nM T55959 CA2HN0 44429214 Ki = 239000 nM T55959 CE30YG 44429218 Ki = 515 nM T55959 CM5HG8 44429219 Ki = 2200 nM T55959 C4I1GO 44429221 Ki = 3780 nM T55959 CDGP34 44429222 Ki = 392000 nM T55959 CW7L3V 44429226 Ki = 810 nM T55959 CKF60U 44429227 Ki = 11000 nM T55959 CX4EM1 44429392 Ki = 830000 nM T55959 C3JNX9 44429393 Ki = 766000 nM T55959 CH9W4Z 44429395 Ki = 1180000 nM T55959 C3O9DN 44429396 Ki = 975000 nM T55959 CO29HT 44429397 Ki = 569000 nM T55959 C75HYO 44429399 Ki = 222000 nM T55959 C7TXV4 44429400 Ki = 313000 nM T55959 CBR73H 44429401 Ki = 1140000 nM T55959 CG9N0T 44429402 Ki = 884000 nM T55959 CQG41A 44430844 IC50 > 10000 nM T55959 CF4BK0 44430849 IC50 = 80 nM T55959 C82VMO 44430851 IC50 = 290 nM T55959 C6CD3M 44431728 Ki = 6.42 nM T55959 CT2UJ0 44431732 Ki = 11.47 nM T55959 CE2QP4 44431734 Ki = 2.25 nM T55959 CHR6F7 44431736 Ki = 10.09 nM T55959 CH6B3Y 44431739 Ki = 2.26 nM T55959 CF42IC 44434165 Ki = 400 nM T55959 CC1R9F 44434885 Ki = 232000 nM T55959 CU5PW7 44434887 Ki = 56000 nM T55959 C0FZ6I 44434888 Ki = 32200 nM T55959 CZ3RM2 44435219 Ki = 6600 nM T55959 C50ZDW 44439863 Ki = 102 nM T55959 CZ9F1A 44440497 Ki = 503 nM T55959 CF8K5H 44441067 Ki = 107 nM T55959 C6P8RJ 44441332 IC50 = 44 nM T55959 CDEY23 44441334 IC50 = 206 nM T55959 COBN96 44441335 IC50 = 125 nM T55959 C23BGW 44441336 IC50 = 122 nM T55959 C92ABN 44441338 IC50 = 1470 nM T55959 C6K8ZB 44441339 IC50 = 1600 nM T55959 CJ2S0W 44441340 IC50 > 4000 nM T55959 C1R0DN 44441341 IC50 = 727 nM T55959 C9FB6Y 44441345 IC50 = 115 nM T55959 CZ34LI 44441346 IC50 = 196 nM T55959 C2GAV7 44441348 IC50 > 4000 nM T55959 CWH92R 44441349 IC50 = 968 nM T55959 C61VKY 44441350 IC50 > 4000 nM T55959 CF4A8D 44441351 IC50 = 1200 nM T55959 CD30KT 44441353 IC50 = 1190 nM T55959 C8ZJU5 44443873 Ki = 11000 nM T55959 C4X5GY 44443875 Ki = 58000 nM T55959 CI0Q6D 44443877 Ki = 94000 nM T55959 COC4G7 44443878 Ki = 9000 nM T55959 C9JB8C 44443887 Ki = 70 nM T55959 C3Q8RJ 44443888 Ki = 6400 nM T55959 CCP50E 44443889 Ki = 830 nM T55959 CSF8J3 44443890 Ki = 140 nM T55959 CRB6J3 44443891 Ki = 30 nM T55959 C0EI1N 44443892 Ki = 12000 nM T55959 CZUT06 44443893 Ki = 2600 nM T55959 CWB8E6 44443894 Ki = 300 nM T55959 CDW62E 44443895 Ki = 500 nM T55959 CR1AP8 44443896 Ki = 3400 nM T55959 CVK42D 44443897 Ki = 170 nM T55959 CEI6Y9 44443898 Ki = 220 nM T55959 C2WC8G 44443899 Ki = 400 nM T55959 C03MYS 44443900 Ki = 1500 nM T55959 C6FY0T 44444517 IC50 = 33000 nM T55959 CMEO07 44444525 IC50 = 8700 nM T55959 C92VUT 44444530 IC50 = 12000 nM T55959 CG0TP9 44444534 IC50 = 2400 nM T55959 CCMZ42 44444540 IC50 = 1100 nM T55959 C0YOW4 44448355 IC50 > 10000 nM T55959 CZS5L9 44448356 IC50 > 10000 nM T55959 CG4D7J 44448357 IC50 > 10000 nM T55959 C9RJX0 44448358 IC50 = 6900 nM T55959 C7AW4C 44448387 IC50 > 10000 nM T55959 C15HXQ 44448388 IC50 > 10000 nM T55959 C1OQ2Y 44448389 IC50 > 10000 nM T55959 CE80KR 44448391 IC50 > 10000 nM T55959 CQV39U 44448392 IC50 > 10000 nM T55959 CPV4Z3 44448423 IC50 > 10000 nM T55959 CFC8I2 44448425 IC50 > 10000 nM T55959 CM8QA0 44448426 IC50 > 10000 nM T55959 C1LIQ2 44448427 IC50 = 8300 nM T55959 CW51IM 44448465 IC50 > 10000 nM T55959 C1MIQ3 44448466 IC50 > 10000 nM T55959 CO4GZ7 44448467 IC50 > 10000 nM T55959 COE35W 44448468 IC50 > 10000 nM T55959 C5GTQ1 44448470 IC50 > 10000 nM T55959 CJ8X7A 44448508 IC50 > 10000 nM T55959 CKO0F9 44448509 IC50 > 10000 nM T55959 C36MOD 44448511 IC50 > 10000 nM T55959 CCR7Q2 44448512 IC50 = 2400 nM T55959 CPS91V 44448544 IC50 > 10000 nM T55959 CO9U4F 44448545 IC50 > 10000 nM T55959 CM6W2E 44448546 IC50 > 10000 nM T55959 CWA0E4 44448547 IC50 = 6300 nM T55959 C9HVB8 44448548 IC50 > 10000 nM T55959 CSYB74 44448582 IC50 > 10000 nM T55959 CF0ZG2 44448584 IC50 > 10000 nM T55959 C3RMF8 44449236 IC50 = 1680 nM T55959 C2UQI1 44449238 IC50 = 1970 nM T55959 CQN4Z9 44449267 IC50 = 3230 nM T55959 CZ3UA5 44449268 IC50 > 34000 nM T55959 CS6R9X 44449270 Ki = 4350 nM T55959 CKH31F 44449272 IC50 > 38000 nM T55959 CGK7O1 44449297 IC50 = 10200 nM T55959 C2O9KI 44449307 IC50 > 10000 nM T55959 CJC38Z 44449333 IC50 > 4000 nM T55959 C6X4JZ 44449340 IC50 > 10000 nM T55959 CCB54W 44449341 IC50 > 10000 nM T55959 C1CPD4 44449368 IC50 = 6300 nM T55959 CR4OB8 44449369 IC50 > 10000 nM T55959 C7W4XU 44449370 IC50 > 10000 nM T55959 CC2ZK5 44449371 IC50 > 10000 nM T55959 CZSE46 44449372 IC50 > 10000 nM T55959 CZY4G7 44449373 IC50 = 1300 nM T55959 CH48QG 44449395 IC50 > 10000 nM T55959 C2YG0E 44449396 IC50 = 2900 nM T55959 CD9LA2 44449397 IC50 > 10000 nM T55959 CWG79A 44449398 IC50 > 10000 nM T55959 CW98KH 44449399 IC50 > 10000 nM T55959 CYM7I3 44449400 IC50 = 4300 nM T55959 CK9UP5 44449401 IC50 > 10000 nM T55959 C8EJ1M 44449434 IC50 > 10000 nM T55959 C6KR7N 44449435 IC50 > 10000 nM T55959 C59NSQ 44449436 IC50 > 10000 nM T55959 C2QF0K 44449437 IC50 = 4500 nM T55959 C2Z6IM 44449438 IC50 > 10000 nM T55959 CJL4G7 44449462 IC50 > 10000 nM T55959 C50SKP 44449464 IC50 > 10000 nM T55959 CT76PB 44449465 IC50 = 3900 nM T55959 COU68C 44449519 IC50 > 10000 nM T55959 C0X2RW 44449521 IC50 > 10000 nM T55959 CG2AD9 44449552 IC50 > 10000 nM T55959 CY0B5K 44449554 IC50 = 3600 nM T55959 CHA59Q 44449589 IC50 = 640 nM T55959 CDQ89E 44449590 IC50 > 10000 nM T55959 C53EYA 44449619 IC50 > 10000 nM T55959 CUXK25 44449620 IC50 = 4300 nM T55959 C7KZ5C 44449623 IC50 > 10000 nM T55959 CZ1L4G 44449624 IC50 > 10000 nM T55959 C8K3XF 44449625 IC50 > 10000 nM T55959 CYRM03 44449651 IC50 > 10000 nM T55959 C15DIZ 44449652 IC50 > 10000 nM T55959 CWO0H5 44449656 IC50 > 10000 nM T55959 C41WXJ 44449718 IC50 = 2430 nM T55959 C2QP0Z 44449729 IC50 > 10000 nM T55959 C3FP2I 44449792 Ki = 3080 nM T55959 C83ICG 44449794 Ki = 1790 nM T55959 CS9ZO8 44449911 Ki = 1540 nM T55959 C50ZLO 44449944 Ki > 10000 nM T55959 CW9P8L 44450088 Ki = 1650 nM T55959 C35FRM 44450119 Ki = 10800 nM T55959 C4AUT7 44450121 Ki = 1090 nM T55959 C52HPA 44450154 Ki = 5750 nM T55959 C9SB0X 44450155 Ki = 420 nM T55959 CAW6S7 44450181 Ki = 380 nM T55959 C4M0PG 44450184 Ki = 950 nM T55959 C4KE7B 44450185 Ki = 2600 nM T55959 C4VL3W 44450211 Ki = 1170 nM T55959 CSQR06 44450212 Ki = 760 nM T55959 CXR4G1 44450213 Ki = 1250 nM T55959 CTX1Q7 44452747 Ki = 4060 nM T55959 CIS3J5 44452748 Ki = 2390 nM T55959 COAL13 44452772 Ki = 4800 nM T55959 C42KFD 44452774 Ki = 2280 nM T55959 CGR0B6 44452775 Ki = 2660 nM T55959 C80CWR 44452935 Ki = 2640 nM T55959 CY01KA 44452990 Ki = 2250 nM T55959 C8Q7OP 44452992 Ki = 1980 nM T55959 CV92RP 44452994 Ki = 2880 nM T55959 CLSI34 44453016 Ki = 1160 nM T55959 CKZN93 44453017 Ki = 2130 nM T55959 CB1OY5 44453042 Ki = 834 nM T55959 C2HFJ7 44453043 Ki = 1930 nM T55959 CY38AM 44453067 Ki = 1750 nM T55959 CBP25X 44453068 Ki = 1410 nM T55959 CR4F7O 44453093 Ki = 1520 nM T55959 C01QKJ 44453119 Ki = 2150 nM T55959 CB06JG 44454485 IC50 > 10000 nM T55959 CISA76 44454488 IC50 > 10000 nM T55959 CE1X7O 44454489 IC50 > 10000 nM T55959 CYRU93 44454493 IC50 > 10000 nM T55959 CKJ2D3 44454526 IC50 > 10000 nM T55959 CB9M0F 44454528 IC50 > 10000 nM T55959 CYCB65 44454556 IC50 > 10000 nM T55959 CH4JN9 44454557 IC50 = 2400 nM T55959 CJB41D 44454559 IC50 > 10000 nM T55959 CQ87FZ 44454585 IC50 > 10000 nM T55959 C8LR9P 44454660 IC50 > 10000 nM T55959 C3T5HK 44454663 IC50 > 10000 nM T55959 C89SJY 44454690 IC50 = 4600 nM T55959 CYZ39A 44454694 IC50 > 10000 nM T55959 C0QVN8 44454719 IC50 > 10000 nM T55959 C01XOI 44454744 IC50 > 10000 nM T55959 C1H0FI 44454746 IC50 = 6200 nM T55959 C43QBZ 44454747 IC50 > 10000 nM T55959 CEY3T6 44454767 IC50 > 10000 nM T55959 C8FBC2 44454794 IC50 > 10000 nM T55959 CJBD47 44454795 IC50 > 10000 nM T55959 C4WOL9 44454797 IC50 > 10000 nM T55959 CU49TR 44454860 IC50 = 7400 nM T55959 COX3W0 44454862 IC50 = 4600 nM T55959 CQF13W 44454863 IC50 > 10000 nM T55959 CU21QR 44454893 IC50 > 10000 nM T55959 CU8K7O 44454894 IC50 > 10000 nM T55959 CVU57D 44454896 IC50 > 10000 nM T55959 C1P5VQ 44454931 IC50 > 10000 nM T55959 CZ2X0T 44454932 IC50 > 10000 nM T55959 CZL97F 44455426 Ki > 10000 nM T55959 CC09EJ 44455512 Ki = 770 nM T55959 C6YQU9 44455589 IC50 = 47 nM T55959 C9PG3H 44455590 IC50 = 320 nM T55959 C1BR2G 44455619 IC50 = 387 nM T55959 CO1X6Z 44455620 IC50 = 172 nM T55959 C8F5CI 44455622 IC50 = 2820 nM T55959 C0EM9R 44455651 IC50 = 138 nM T55959 CW7E6X 44455652 IC50 = 275 nM T55959 C3W1EZ 44455653 IC50 = 3010 nM T55959 CI4K0E 44455654 IC50 = 1210 nM T55959 CZV45C 44455655 IC50 = 800 nM T55959 C0L9YB 44455677 IC50 = 21000 nM T55959 CV10IJ 44455678 IC50 = 15700 nM T55959 CK47LB 44455681 IC50 > 40000 nM T55959 CR24HA 44455708 IC50 = 5950 nM T55959 CJM9O8 44455710 IC50 = 6510 nM T55959 COV02B 44455738 IC50 = 2130 nM T55959 C3CXW8 44455739 IC50 = 3780 nM T55959 CO4B1F 44455740 IC50 = 19600 nM T55959 C3I6TO 44455742 IC50 = 421 nM T55959 C76JRV 44455761 IC50 = 194 nM T55959 CSX82U 44455763 IC50 = 2730 nM T55959 C16SFL 44455822 Ki = 2500 nM T55959 C8MV5J 44455895 IC50 = 67 nM T55959 CAB61T 44455930 IC50 = 11 nM T55959 CD90LW 44456110 IC50 = 28 nM T55959 C2K8HO 44456196 IC50 = 12 nM T55959 C08MBY 44456312 Ki = 330 nM T55959 CMT7G2 44456313 IC50 = 115 nM T55959 C12XGE 44456400 Ki > 10000 nM T55959 CI8HF6 44456422 IC50 = 8 nM T55959 CVTY18 44456425 IC50 = 31 nM T55959 CB68FX 44456464 IC50 = 55 nM T55959 C8TPF7 44456465 IC50 = 2960 nM T55959 C6SL0P 44456466 IC50 = 1540 nM T55959 CS74YL 44457050 Ki > 30000 nM T55959 C36OQY 44457051 Ki > 10000 nM T55959 CKI8L5 44457058 Ki > 3000 nM T55959 CQS23B 44457059 Ki > 6000 nM T55959 CC9ZF1 44462051 Ki = 0.48 nM T55959 CN3H5R 44462082 IC50 = 1.7 nM T55959 CL9O8M 44462783 IC50 = 71 nM T55959 C91PCM 44466344 Ki = 31.62 nM T55959 CZA36I 44466345 Ki = 25.12 nM T55959 C63XKS 44467026 Ki = 79.43 nM T55959 CH4WM3 44467027 Ki = 79.43 nM T55959 C3T4BX 44467028 Ki = 125.89 nM T55959 CG4R7A 44467101 Ki = 251.19 nM T55959 CW2K9E 44467103 Ki = 501.19 nM T55959 CL0JR9 44467104 Ki = 794.33 nM T55959 C4CX9E 44467173 Ki = 1584.89 nM T55959 CG4H1R 44467174 Ki = 501.19 nM T55959 CLU6A0 44467177 Ki = 79.43 nM T55959 C4RBV8 44467889 Ki = 50.12 nM T55959 CJB37C 44467892 Ki = 158.49 nM T55959 CF4ZM8 44467957 Ki = 50.12 nM T55959 CTO9R8 44467960 Ki = 199.53 nM T55959 C4DL5C 44469677 IC50 > 10000 nM T55959 C5N4KE 44472633 IC50 = 4800 nM T55959 CM6Q7W 44474580 Ki = 586 nM T55959 C73XSD 44474582 Ki = 1910 nM T55959 C68VDK 44474583 Ki = 913 nM T55959 C21WPR 44474586 Ki = 223 nM T55959 C3DHG0 44511399 IC50 = 116 nM T55959 CU9MO1 44539110 IC50 = 19.95 nM T55959 CAL8V3 44539203 Ki = 50.12 nM T55959 CO1E5C 44539964 IC50 = 1240 nM T55959 CLMY52 44539967 IC50 = 58 nM T55959 CLO73R 44540428 IC50 = 616 nM T55959 CV92IJ 44541354 IC50 = 3.7 nM T55959 C5Q3NI 44542504 IC50 > 100 nM T55959 C5F1UC 44542505 Ki > 10000 nM T55959 CYX7H5 44542510 IC50 = 410 nM T55959 C71QGD 44542511 IC50 > 100 nM T55959 C8V7UL 44542657 Ki = 140 nM T55959 C6ECJ1 44542658 IC50 = 258 nM T55959 C2EDU6 44542955 IC50 > 100 nM T55959 CTW5I9 44542956 Ki > 10000 nM T55959 C03MXJ 44543264 IC50 = 7978 nM T55959 CL5UK7 44543265 IC50 = 950 nM T55959 CBL30Z 44543269 Ki = 1700 nM T55959 CHIY92 44543270 Ki > 10000 nM T55959 C1YIC9 44560434 IC50 = 1.86 nM T55959 C7G9WM 44560436 IC50 = 6.45 nM T55959 C35XEU 44560438 IC50 = 6.42 nM T55959 CBTX17 44560440 IC50 = 8.74 nM T55959 CB0K6T 44560442 IC50 = 111 nM T55959 CWCT08 44560444 IC50 = 76 nM T55959 C69ETG 44560446 IC50 = 68.7 nM T55959 CK2PD5 44560493 IC50 = 4.09 nM T55959 C2SZ1B 44560495 IC50 = 13 nM T55959 C9U5SE 44560498 IC50 = 3.93 nM T55959 CNK4F6 44560500 IC50 = 65.7 nM T55959 CU05HZ 44560502 IC50 = 135 nM T55959 C87VZD 44560504 IC50 = 173 nM T55959 CV0BF4 44560506 IC50 = 81.6 nM T55959 CS9N0U 44560575 IC50 = 4000 nM T55959 CYNS29 44560577 IC50 = 5000 nM T55959 CF5BX9 44560599 IC50 = 119 nM T55959 CNF81T 44560602 IC50 = 8.6 nM T55959 CWB6S3 44560604 IC50 = 5.9 nM T55959 CJQ4R5 44560606 IC50 = 17.5 nM T55959 C7TO9F 44560608 IC50 = 22.2 nM T55959 C17ZEN 44560622 IC50 > 10000 nM T55959 CN1K6R 44560623 IC50 = 2400 nM T55959 C9BV0O 44560624 IC50 = 7000 nM T55959 CY72NM 44560625 IC50 > 10000 nM T55959 C0FW5J 44560626 IC50 = 4600 nM T55959 CLW2R6 44560627 IC50 = 10000 nM T55959 CI1XD4 44560628 IC50 > 10000 nM T55959 C1NCT4 44560653 IC50 = 22.1 nM T55959 C8MPN0 44560655 IC50 = 6.9 nM T55959 CWG57V 44560657 IC50 = 6.1 nM T55959 CH79ZT 44560659 IC50 = 9.6 nM T55959 C51DKQ 44560671 IC50 = 2500 nM T55959 CBMT59 44560672 IC50 = 2500 nM T55959 C1R8PQ 44560673 IC50 > 10000 nM T55959 CGK29S 44560675 IC50 = 180 nM T55959 CG4YN5 44560676 IC50 = 3400 nM T55959 CNM1Q6 44560708 IC50 > 10000 nM T55959 CG6FL1 44560709 IC50 = 4500 nM T55959 CL9J2E 44560710 IC50 > 10000 nM T55959 C36IOW 44560711 IC50 = 6000 nM T55959 CLM2F8 44560712 IC50 = 1000 nM T55959 C3OG8F 44560713 IC50 = 1000 nM T55959 C9B5CE 44560714 IC50 = 1000 nM T55959 CP7RQ8 44562623 IC50 > 10000 nM T55959 CHE68Z 44562624 IC50 > 10000 nM T55959 CR4TG7 44562625 IC50 = 4000 nM T55959 CH32FI 44562626 IC50 = 10000 nM T55959 CX1P3L 44562627 IC50 > 10000 nM T55959 C0S8ZG 44562682 IC50 > 10000 nM T55959 C2HKE0 44562772 IC50 > 10000 nM T55959 C50WKO 44562773 IC50 = 3500 nM T55959 C3JD7Y 44562774 IC50 = 8000 nM T55959 CS0LD7 44562775 IC50 = 3000 nM T55959 C7AC8Z 44562776 IC50 = 5000 nM T55959 CU6G4W 44562777 IC50 > 10000 nM T55959 CCA0H2 44562815 IC50 > 10000 nM T55959 CQ0I5R 44562816 IC50 = 4000 nM T55959 CC1IF3 44562817 IC50 = 5000 nM T55959 CR28PD 44563213 IC50 = 10000 nM T55959 CU4PD5 44563214 IC50 = 1600 nM T55959 CGKL94 44563257 IC50 = 4700 nM T55959 C8TYL3 44563258 IC50 > 10000 nM T55959 C8XUD6 44563259 IC50 > 10000 nM T55959 CIG6Z4 44563260 IC50 > 10000 nM T55959 C9VFW6 44563261 IC50 > 10000 nM T55959 C9N0RT 44563646 Ki = 87.6 nM T55959 CEG7S1 44563647 Ki = 35.5 nM T55959 C41KWG 44563667 Ki = 179.7 nM T55959 CI6A1Q 44563668 Ki = 118.7 nM T55959 CL83PU 44563669 Ki = 274 nM T55959 CJD73U 44565305 IC50 = 5340 nM T55959 CM8LR1 44568174 IC50 > 10000 nM T55959 CCRI61 44568175 IC50 = 6400 nM T55959 CB3VF8 44568176 IC50 = 6400 nM T55959 C6T2BK 44568293 IC50 = 4200 nM T55959 CA1NJ9 44568294 IC50 = 16000 nM T55959 CA21KI 44568295 IC50 = 6100 nM T55959 CX50DP 44568296 IC50 = 105 nM T55959 COB14G 44568297 IC50 = 260 nM T55959 C3I6FM 44568320 IC50 = 85 nM T55959 C4QYH2 44568321 IC50 = 200 nM T55959 CKT30F 44568322 IC50 > 10000 nM T55959 C1HA7U 44568323 IC50 > 10000 nM T55959 C9CJP2 44568324 IC50 > 10000 nM T55959 C81XJM 44568325 IC50 = 6900 nM T55959 CVA67X 44568347 Ki = 6000 nM T55959 C3SW7N 44568349 IC50 = 3800 nM T55959 CLTG36 44568350 IC50 = 1500 nM T55959 C9MNC0 44568351 IC50 = 3600 nM T55959 CB58VS 44568378 IC50 > 10000 nM T55959 CYN68I 44568379 IC50 > 10000 nM T55959 CY3NQ8 44568652 IC50 = 2000 nM T55959 C02GHU 44568653 IC50 = 320 nM T55959 C8HNK7 44568691 IC50 = 2100 nM T55959 C7FBU8 44568693 IC50 = 5900 nM T55959 CD48SQ 44568694 IC50 = 11000 nM T55959 CSZ7V2 44568750 IC50 = 2800 nM T55959 CWG32I 44572166 Ki > 10000 nM T55959 C97VKX 44572751 Ki = 2115 nM T55959 CJ1VI8 44572802 Ki = 5400 nM T55959 CU25XD 44572810 Ki = 3261 nM T55959 C6S4IO 44576826 IC50 = 0.23 nM T55959 C7WO9Z 44576828 IC50 = 0.32 nM T55959 CE5JC1 44576830 IC50 = 3.6 nM T55959 C4XBZ0 44576832 IC50 = 1.4 nM T55959 COT0K9 44576862 IC50 = 11 nM T55959 CYXV83 44576864 IC50 = 3.6 nM T55959 CS4XT1 44576866 IC50 = 0.8 nM T55959 CCB06N 44576868 IC50 = 0.8 nM T55959 CV45DH 44576870 IC50 = 0.9 nM T55959 C42FLK 44576888 IC50 = 2.2 nM T55959 COP7S3 44576890 IC50 = 8 nM T55959 C4ISW9 44576892 IC50 = 47 nM T55959 CC0A8W 44578263 Ki = 3410 nM T55959 CY40JQ 44578265 Ki = 4190 nM T55959 CFJB16 44578266 Ki = 2670 nM T55959 CE54ZK 44578267 Ki = 2760 nM T55959 CSFE81 44578268 Ki = 2070 nM T55959 CQ30GC 44578271 Ki = 2910 nM T55959 C8HB0Z 44578272 Ki = 2390 nM T55959 CV63SW 44578313 Ki = 1380 nM T55959 CH3U5D 44578314 Ki = 2700 nM T55959 C8XAO4 44578315 Ki = 2080 nM T55959 CS70JE 44578316 Ki = 2890 nM T55959 CAP14F 44578317 Ki = 2950 nM T55959 CUVQ89 44578318 Ki = 2550 nM T55959 C17YVO 44578319 Ki = 2690 nM T55959 CPQC54 44578368 Ki = 2130 nM T55959 CTE6V8 44578370 Ki = 2010 nM T55959 C4VO1L 44578371 Ki = 3340 nM T55959 CXZ05B 44578372 Ki = 3210 nM T55959 C8AP4K 44578374 Ki = 1900 nM T55959 CDMH40 44578375 Ki = 2970 nM T55959 CUQV50 44579565 IC50 = 13 nM T55959 CS91HK 44579613 IC50 > 10 nM T55959 C0KBZ4 44580189 Ki > 1000 nM T55959 C2U7TG 44580702 Ki > 1000 nM T55959 C0S4IO 44580703 Ki > 2000 nM T55959 C3ONV6 44580704 Ki > 1000 nM T55959 CRCH48 44582675 Ki > 10000 nM T55959 CEJ4R8 44582676 Ki > 10000 nM T55959 C5QB4K 44582678 Ki > 10000 nM T55959 C3L5ER 44583033 IC50 = 1.2 nM T55959 CWK97I 44584916 IC50 = 199526.23 nM T55959 CBIO97 44585469 IC50 = 0.05 ug.mL-1 T55959 C4HJE6 44586246 Ki = 1485 nM T55959 CXKQ61 44587384 IC50 > 10000 nM T55959 CZLV68 44587385 IC50 = 7500 nM T55959 C8SFJ1 44587386 IC50 > 10000 nM T55959 CPBR52 44587387 IC50 > 10000 nM T55959 C4D7GP 44587388 IC50 > 10000 nM T55959 CRL0H9 44587389 IC50 = 4000 nM T55959 C5PV7Q 44587390 IC50 > 10000 nM T55959 C5IUL8 44587443 IC50 > 10000 nM T55959 C59KDV 44587445 IC50 > 10000 nM T55959 CLCE75 44587446 IC50 > 10000 nM T55959 CPF01B 44587447 IC50 > 10000 nM T55959 CIL89C 44587448 IC50 = 7000 nM T55959 CF0I6D 44587449 IC50 = 10000 nM T55959 C0J4LS 44587450 IC50 = 2600 nM T55959 CZVX16 44587463 IC50 > 10000 nM T55959 C6UI9D 44587464 IC50 > 10000 nM T55959 C6YQS2 44587465 IC50 = 5700 nM T55959 CNV4I9 44587466 IC50 > 10000 nM T55959 CL10BT 44587467 IC50 = 4000 nM T55959 CX5KZ1 44587468 IC50 > 10000 nM T55959 C0OYJ4 44587469 IC50 > 10000 nM T55959 C2HUA1 44587470 IC50 > 10000 nM T55959 CIW41M 44587471 IC50 > 10000 nM T55959 CCKE83 44587472 IC50 > 10000 nM T55959 C4SGR3 44587473 IC50 > 10000 nM T55959 C47OBV 44587474 IC50 > 10000 nM T55959 CQ79SU 44587475 IC50 = 1400 nM T55959 CUE9C6 44587476 IC50 > 10000 nM T55959 C37ZEB 44587477 IC50 > 10000 nM T55959 CY0F1M 44587482 IC50 = 3800 nM T55959 CL5M2J 44587483 IC50 > 10000 nM T55959 CRN0Z1 44587484 IC50 > 10000 nM T55959 CTN0Q1 44587485 IC50 > 10000 nM T55959 CAHW83 44587486 IC50 > 10000 nM T55959 CJY60H 44587487 IC50 > 10000 nM T55959 C3OL1M 44587488 IC50 > 10000 nM T55959 C56QTZ 44587489 IC50 > 10000 nM T55959 CD60KY 44587995 IC50 = 92 nM T55959 CZ98JO 44587997 IC50 = 16 nM T55959 CAXU48 44587999 IC50 = 47 nM T55959 C6FPZ9 44588001 IC50 = 92 nM T55959 C8F7IT 44588013 IC50 = 170 nM T55959 C8LUE2 44588015 IC50 = 1300 nM T55959 C7Y4QV 44588017 IC50 = 14 nM T55959 C5JQY4 44588019 IC50 = 6 nM T55959 C62JSH 44588021 IC50 = 13 nM T55959 C43ODT 44588187 IC50 = 0.82 nM T55959 CKPE78 44588189 IC50 = 6.5 nM T55959 C57QYV 44588191 IC50 = 42 nM T55959 CPR9K4 44588193 IC50 = 7 nM T55959 CLIV63 44588195 IC50 = 6 nM T55959 CN6RC7 44588197 IC50 = 3.3 nM T55959 CH18RV 44588223 IC50 = 15 nM T55959 CXA2D6 44588225 IC50 = 2.5 nM T55959 C4RZ1U 44588227 IC50 = 102 nM T55959 CQSC48 44588229 IC50 = 18 nM T55959 C4WB1N 44589201 Ki = 1260 nM T55959 C69KAB 44590643 IC50 > 10000 nM T55959 CLQ2N4 44590644 IC50 > 10000 nM T55959 CJ2D4T 44590690 Ki = 27240 nM T55959 C0RHT8 44590691 IC50 = 38440 nM T55959 CQCG57 44590692 IC50 = 8555 nM T55959 CS7H9U 44590693 Ki = 30320 nM T55959 C38PUH 44590694 Ki = 6500 nM T55959 CDB8Z5 44590725 Ki = 16370 nM T55959 C0N5RO 44590726 Ki = 7328 nM T55959 C4H6PT 44590727 Ki = 4576 nM T55959 C3TUD7 44590728 Ki = 3868 nM T55959 CNL38Q 44590729 Ki = 3387 nM T55959 C7RBE8 44590819 Ki > 10000 nM T55959 CYBL93 44590820 Ki > 10000 nM T55959 CI6R1Z 44592120 IC50 = 861 nM T55959 C1QO8J 44592121 IC50 = 2100 nM T55959 C7LKH8 44592122 IC50 > 10000 nM T55959 CVT6R5 44592123 IC50 = 19000 nM T55959 C4KM6A 44592153 IC50 > 30000 nM T55959 CV8E7O 44592155 IC50 > 30000 nM T55959 CK47SV 44592156 IC50 = 3000 nM T55959 C4W1XJ 44592157 IC50 = 66 nM T55959 CMS5I2 44592158 IC50 = 7700 nM T55959 CSU06J 44592195 IC50 = 88 nM T55959 CZ6L3I 44592196 IC50 = 210 nM T55959 CJO9K5 44592245 IC50 > 31000 nM T55959 CQ12YR 44593444 IC50 = 140 nM T55959 CPH6S0 44593451 IC50 = 3500 nM T55959 C30HFZ 44593522 IC50 = 7100 nM T55959 CI3T5N 44593629 Ki = 17 nM T55959 C1DI5Z 44593686 IC50 > 10000 nM T55959 C7YLS4 44593687 IC50 = 3400 nM T55959 C6KGF2 44593688 IC50 > 10000 nM T55959 CU8F9L 44593689 IC50 = 4200 nM T55959 CR18ZA 44593690 IC50 > 10000 nM T55959 C20YZD 44593691 IC50 > 10000 nM T55959 CN52LH 44593692 IC50 > 10000 nM T55959 C7IU8S 44593694 IC50 = 2500 nM T55959 C9SM4D 44593695 IC50 = 4100 nM T55959 CSQ14O 44593696 IC50 > 10000 nM T55959 CI10GR 44610722 IC50 > 28000 nM T55959 CW84TH 44610723 IC50 = 4900 nM T55959 CPIB93 44610724 IC50 = 2800 nM T55959 CVR29I 44625567 Ki = 31.62 nM T55959 C24WVM 44625568 Ki = 100 nM T55959 COM81X 44625569 Ki = 7.943 nM T55959 CR8I3P 44625570 Ki = 158.49 nM T55959 C2D0TJ 44625571 Ki = 158.49 nM T55959 C6LD5P 44625653 Ki = 501.19 nM T55959 CND19I 45102009 IC50 = 346 nM T55959 CW0RU3 45102635 Ki > 6460 nM T55959 CXJ6A2 45140180 IC50 = 20927 nM T55959 CT6XO9 45140370 IC50 = 22834 nM T55959 C7MB5N 45141377 IC50 = 3620 nM T55959 CMSH89 45141378 IC50 > 100 nM T55959 CTL0U6 45141609 IC50 > 100 nM T55959 CB9QZ6 45263405 IC50 = 1600 nM T55959 CP3S0Q 45266826 EC50 = 49.1 nM T55959 CPGO97 45267145 IC50 = 7830 nM T55959 CTL3Z5 45267156 IC50 > 4000 nM T55959 C5DGO1 45267167 IC50 = 644 nM T55959 CP7XE6 45267597 Ki > 10000 nM T55959 CK58HY 45267611 Ki > 3160 nM T55959 C3D9TN 45267621 Ki > 1584.89 nM T55959 CGR34K 45267873 Ki = 28 nM T55959 CEWR12 45268018 IC50 = 1070 nM T55959 CRP90V 45268466 Ki = 2680 nM T55959 CSJ4L2 45268478 Ki = 3130 nM T55959 CQJ9X1 45268495 Ki = 39.81 nM T55959 CO2X9T 45268882 IC50 > 40000 nM T55959 C71XIB 45268898 IC50 = 1270 nM T55959 CHP12M 45268914 IC50 = 36 nM T55959 CUQ23Z 45268922 IC50 = 1060 nM T55959 C5OED7 45269318 Ki = 1360 nM T55959 CF2P9H 45269325 Ki > 10000 nM T55959 CQ03ZU 45269337 Ki > 10000 nM T55959 CXE36D 45269351 Ki > 10000 nM T55959 CVA9E0 45269726 IC50 > 2920 nM T55959 CS0Z8C 45269735 IC50 > 4000 nM T55959 CL6W3X 45269754 IC50 = 60 nM T55959 CL1XW2 45270129 Ki = 12.02 nM T55959 CX31KD 45270149 Ki > 10000 nM T55959 C3GA6N 45270158 Ki = 2040 nM T55959 C3KI7Q 45270163 Ki > 10000 nM T55959 C0QR1E 45270171 Ki > 10000 nM T55959 C6YI5N 45270172 Ki > 10000 nM T55959 CZ9DA3 45270173 Ki = 3470 nM T55959 C13GPD 45270570 IC50 = 480 nM T55959 C0HV4C 45270577 IC50 = 353 nM T55959 COFD89 45270589 IC50 = 6 nM T55959 CEX26T 45270595 IC50 = 200 nM T55959 C13QSU 45270993 Ki = 2650 nM T55959 CU9HV3 45271001 Ki = 3720 nM T55959 C71AON 45271011 Ki > 10000 nM T55959 CI01KJ 45271024 Ki = 3981.07 nM T55959 C62UVG 45271383 IC50 > 4000 nM T55959 C61TGI 45271390 IC50 = 1600 nM T55959 C1S6TI 45271840 Ki = 2340 nM T55959 C3QAP5 45271853 Ki = 3110 nM T55959 CFG5Z3 45271864 Ki > 10000 nM T55959 C3AJ7I 45271873 Ki = 501.19 nM T55959 CT04SP 45271883 Ki = 31.62 nM T55959 C1G9IK 45272302 IC50 = 330 nM T55959 CPM1U3 45272720 Ki = 3440 nM T55959 C4VAE9 45272734 Ki = 4100 nM T55959 CRUN86 45273003 Ki = 78 nM T55959 C4P1FO 45273132 IC50 = 400 nM T55959 CUK91L 45273154 IC50 = 270 nM T55959 C5LB6F 45273161 IC50 = 3470 nM T55959 CT3V0B 45273663 Ki = 2750 nM T55959 CINR73 45273666 Ki = 3470 nM T55959 C3Q0GZ 45273673 Ki > 3160 nM T55959 CZU06K 45273676 Ki = 199.53 nM T55959 CQS5X0 45378248 Ki = 79.43 nM T55959 C7C9HW 45378386 Ki = 5.012 nM T55959 C51WBF 45378387 Ki = 6.31 nM T55959 CS04YD 45379827 Ki = 457.09 nM T55959 CMU6Z8 45379828 Ki = 56.23 nM T55959 C1SCJ9 45379829 Ki = 660.69 nM T55959 CK6L2S 45379946 Ki = 25.12 nM T55959 CNQT48 45379947 Ki = 12.59 nM T55959 C5TQ8X 45379948 Ki = 501.19 nM T55959 CP82MH 45379949 Ki = 19.95 nM T55959 CNSK69 45379950 Ki = 50.12 nM T55959 CM61UN 45380063 Ki = 251.19 nM T55959 C97ZQE 45380064 Ki = 100 nM T55959 CEFO86 45380065 Ki = 19.95 nM T55959 C53JYC 45380066 Ki = 79.43 nM T55959 C46FLB 45380180 Ki = 630.96 nM T55959 C89XTJ 45380181 Ki = 39.81 nM T55959 CYAE52 45380182 Ki = 63.1 nM T55959 C6BLR9 45380183 Ki = 25.12 nM T55959 CO8Z1P 45380184 Ki = 50.12 nM T55959 CE1M3S 45380185 Ki = 79.43 nM T55959 C1OK5Z 45481773 IC50 = 91 nM T55959 CS0W9K 45481774 IC50 > 10000 nM T55959 C5SN4D 45481775 IC50 = 28 nM T55959 CZ02KA 45481776 IC50 = 177 nM T55959 CCOL45 45481778 IC50 = 112 nM T55959 CX68LG 45481779 IC50 = 1200 nM T55959 C52FTP 45481780 IC50 = 71 nM T55959 C0NAE6 45481784 IC50 = 1100 nM T55959 CG75XM 45481786 IC50 = 74 nM T55959 C5F8QK 45481787 IC50 = 9 nM T55959 CQ89WZ 45481788 IC50 = 900 nM T55959 C7BQX4 45481789 IC50 = 232 nM T55959 C1O8ZD 45481790 IC50 = 16 nM T55959 CO1Z4X 45481791 IC50 = 200 nM T55959 CF6R7M 45481792 IC50 = 10.1 nM T55959 CWEK71 45481794 IC50 = 76 nM T55959 C97JBX 45483401 Ki = 1 nM T55959 C9K4XC 45483416 Ki = 659 nM T55959 CZQ6H8 45483429 Ki = 5530 nM T55959 C3HAF8 45483430 Ki = 452 nM T55959 CG2SM9 45483458 Ki = 87 nM T55959 CFM9P8 45483465 Ki = 1360 nM T55959 C5DS3M 45483506 Ki = 470 nM T55959 CHCA47 45483511 Ki > 6000 nM T55959 CI89OX 45487689 IC50 = 1300 nM T55959 CC75GW 45487699 IC50 = 7400 nM T55959 CNFI42 45487726 IC50 > 40000 nM T55959 CAO36Q 45487761 IC50 > 28000 nM T55959 C80FMT 45487762 IC50 > 68000 nM T55959 CL9SM3 45487783 IC50 = 5800 nM T55959 CL1H2W 46200976 Ki = 6976 nM T55959 C79ZBC 46200977 Ki = 3604 nM T55959 CI39BE 46216792 IC50 = 620 nM T55959 CKCN84 46225028 Ki > 10000 nM T55959 C34ZXM 46225029 Ki = 137 nM T55959 CGY19F 46226540 Ki = 2.5 nM T55959 C79GDE 46226541 Ki = 890 nM T55959 C0H7ID 46226542 Ki = 180 nM T55959 C5TSH8 46226543 Ki = 690 nM T55959 CL07MO 46226544 Ki = 21 nM T55959 CMK1Z6 46226545 Ki = 6.6 nM T55959 C1KSD4 46226546 Ki = 20 nM T55959 CED57N 46226547 Ki = 540 nM T55959 C27DWI 46226548 Ki = 690 nM T55959 C3I4ZU 46226549 Ki = 350 nM T55959 C6UDJ2 46226550 Ki = 1300 nM T55959 C8Q0JS 46226551 Ki = 210 nM T55959 C6SGC5 46226552 Ki = 800 nM T55959 C70RNJ 46226553 Ki = 710 nM T55959 C72NRZ 46226554 Ki = 93 nM T55959 C8FM7G 46226555 Ki = 160 nM T55959 CJS97C 46226556 Ki = 230 nM T55959 CB8XA5 46226557 Ki = 16 nM T55959 COC3L5 46226572 Ki = 1 nM T55959 CJKZ16 46226573 Ki = 3.9 nM T55959 CF6I8D 46226574 Ki = 5.5 nM T55959 CE0W4J 46227268 Ki = 857 nM T55959 CY5FD9 46227269 Ki = 4598 nM T55959 CJ9OF6 46228636 Ki = 3.981 nM T55959 CSNI09 46228719 Ki = 125.89 nM T55959 CG68MR 46228720 Ki = 31.62 nM T55959 C5NB2Z 46228786 Ki = 10 nM T55959 C5JPE2 46229669 Ki = 1220 nM T55959 C4B0FX 46229670 Ki = 960 nM T55959 C39VDA 46229671 Ki = 726 nM T55959 CS0EJ4 46229672 Ki = 4186 nM T55959 C32VBR 46229686 Ki > 1000 nM T55959 CN4HT2 46230756 Ki > 6220 nM T55959 C7OB2G 46235733 IC50 = 141.25 nM T55959 CJ2D3O 46701015 IC50 = 123.03 nM T55959 CM04ZI 46701016 IC50 = 47.86 nM T55959 C0JWP5 46701017 IC50 = 147.91 nM T55959 C5H0MJ 46701086 IC50 = 204.17 nM T55959 C9HWI7 46701087 IC50 = 83.18 nM T55959 CVE5O1 46701088 IC50 = 14.13 nM T55959 C1VPM0 46701089 IC50 = 54.95 nM T55959 CQ8B6R 46701090 IC50 = 10 nM T55959 C6C0FS 46701091 IC50 = 25.12 nM T55959 CC0M7T 46830494 IC50 = 1475 nM T55959 C2ZGO0 46830791 IC50 = 2113 nM T55959 CYWA02 46831080 IC50 = 2326 nM T55959 COF0Q6 46831083 IC50 = 2570 nM T55959 CZF25N 46831086 IC50 = 386 nM T55959 CDF9H4 46831389 IC50 = 3185 nM T55959 CL7XJ8 46831392 IC50 = 2086 nM T55959 CEV89K 46831395 IC50 = 2618 nM T55959 C95KSN 46833979 IC50 = 2409 nM T55959 C18CYM 46833983 IC50 = 1872 nM T55959 CUD7M8 46833985 IC50 = 267 nM T55959 CD0PH8 46833987 IC50 = 262 nM T55959 CHPS94 46833989 IC50 = 998 nM T55959 C80NHM 46834258 IC50 = 509 nM T55959 C1GPD3 46834260 IC50 = 5500 nM T55959 C37MDG 46834262 IC50 = 291 nM T55959 CQ7S3X 46837648 IC50 = 61 nM T55959 CL7VN1 46837649 IC50 = 44 nM T55959 CU7OG4 46837651 IC50 = 16000 nM T55959 C5WNL1 46837652 IC50 = 12000 nM T55959 COX2H5 46837653 IC50 = 4200 nM T55959 CWZY17 46837780 IC50 = 285 nM T55959 CV2NT3 46837781 IC50 = 832 nM T55959 CT83MU 46837782 IC50 > 100000 nM T55959 C5TY3Q 46837783 IC50 > 100000 nM T55959 CWJF83 46837784 IC50 = 2140 nM T55959 C0ZSY5 46837785 IC50 = 1020 nM T55959 CBQJ74 46837922 IC50 = 23 nM T55959 C8UWQ2 46837923 IC50 = 30 nM T55959 CCX8T0 46837924 IC50 = 230 nM T55959 CBH49N 46837925 IC50 = 2870 nM T55959 CH76RQ 46855361 Ki = 39.81 nM T55959 CFJ3Q4 46855363 Ki = 1258.93 nM T55959 CEG23T 46855638 Ki = 3.162 nM T55959 CFW0B9 46855640 Ki = 5.012 nM T55959 CKS74N 46855641 Ki = 251.19 nM T55959 C7FPT6 46855642 Ki = 3.981 nM T55959 CZS2G8 46855643 Ki = 100 nM T55959 C9AG3X 46855785 Ki = 100 nM T55959 C2WKY8 46855786 Ki = 501.19 nM T55959 CB51DQ 46855787 Ki = 398.11 nM T55959 CHT1G5 46855789 Ki = 1258.93 nM T55959 CLX6M3 46855790 Ki = 79.43 nM T55959 C0CG4F 46866510 Ki = 12.59 nM T55959 C1OE2K 46877858 IC50 = 2040 nM T55959 C7PDE6 46877860 IC50 = 11700 nM T55959 C89FYG 46877878 IC50 = 265 nM T55959 CT3R2F 46877879 IC50 = 0.76 nM T55959 CK8A1O 46880462 Ki > 10000 nM T55959 C9KDP4 46880463 Ki > 10000 nM T55959 CODR73 46880498 Ki > 10000 nM T55959 CHJ5Y6 46880566 Ki > 10000 nM T55959 CE9PG2 46880567 Ki > 10000 nM T55959 C01PGO 46880568 Ki > 10000 nM T55959 CS7L4X 46880569 Ki > 10000 nM T55959 C0PXY7 46880628 Ki > 10000 nM T55959 CD37LU 46880629 Ki > 10000 nM T55959 CUY89F 46880630 Ki > 10000 nM T55959 C4P6XS 46880631 Ki > 10000 nM T55959 CJ53KF 46880672 Ki > 10000 nM T55959 CYJC08 46880673 Ki > 10000 nM T55959 C1RI9O 46880674 Ki > 10000 nM T55959 CMS27C 46882857 Ki = 945 nM T55959 CM45ZP 46882858 Ki = 501 nM T55959 C3IGF1 46882859 Ki = 2430 nM T55959 CHLZ97 46882860 Ki = 3070 nM T55959 C4B8EX 46882909 Ki = 2070 nM T55959 CFY95C 46882910 Ki = 516 nM T55959 C6GJ1F 46882911 Ki = 2370 nM T55959 C0SQX2 46882912 Ki = 2560 nM T55959 CV94JW 46882937 Ki = 2540 nM T55959 CM5Z4G 46882938 Ki = 3590 nM T55959 CJV6R1 46882939 Ki = 3090 nM T55959 C60YMF 46883462 Ki = 1090 nM T55959 C7J6GU 46883497 Ki = 630 nM T55959 C3F5AS 46883498 Ki = 404 nM T55959 CRSE34 46883499 Ki = 273 nM T55959 C0CX3O 46883500 Ki = 2600 nM T55959 C78FKZ 46888072 IC50 = 30 nM T55959 CH56AN 46890391 Ki > 3160 nM T55959 CPDX34 46890392 Ki = 1390 nM T55959 C0YGP2 46890393 Ki = 1400 nM T55959 C61INJ 46890394 Ki > 3160 nM T55959 CI14SE 46890441 Ki = 6810 nM T55959 CP4GD3 46890442 Ki = 2370 nM T55959 CQI2Y8 46890443 Ki > 3160 nM T55959 CZ2MG7 46890444 Ki > 10000 nM T55959 CP6A8K 46890445 Ki = 4060 nM T55959 CD5J8B 46890446 Ki = 4870 nM T55959 CYK9D2 46890489 Ki > 10000 nM T55959 CCR04L 46890490 Ki = 3460 nM T55959 CT4O9M 46890491 Ki = 1760 nM T55959 CGPM19 46890493 Ki = 4900 nM T55959 C68AJP 46933238 Ki = 0.631 nM T55959 CX7R3H 46933845 Ki > 10000 nM T55959 CAY75I 46934585 Ki = 3.981 nM T55959 C2LZJ0 49783209 Ki = 2020 nM T55959 C57SMG 49783415 Ki > 10000 nM T55959 C0TG6I 49783419 Ki > 10000 nM T55959 CO6W0D 49798171 Ki = 501.19 nM T55959 CHQ7I8 49798172 Ki = 398.11 nM T55959 CMBX16 49798173 Ki = 158.49 nM T55959 CMO8V7 49798193 Ki = 1584.89 nM T55959 C60YCR 49798194 Ki = 100 nM T55959 C85KNS 49798241 Ki = 316.23 nM T55959 CQ4G1V 49798242 Ki = 501.19 nM T55959 C01JNE 49798243 Ki = 39.81 nM T55959 CC6MF8 49798244 Ki = 50.12 nM T55959 CYAS45 49798266 Ki = 1000 nM T55959 C2UO0F 49799236 IC50 > 100000 nM T55959 C6FH8G 49799237 IC50 > 100000 nM T55959 CZ3US5 49799443 Ki = 158.49 nM T55959 CQH0U4 49799522 Ki = 125.89 nM T55959 CZ76MQ 49799633 IC50 = 70 nM T55959 CU28RO 49799634 IC50 = 8250 nM T55959 CN89XG 49799642 IC50 = 10000 nM T55959 C85MBT 49799643 IC50 = 453 nM T55959 CK6IA0 49799933 IC50 > 10000 nM T55959 C58AWR 49818125 Ki = 1.514 nM T55959 CDV79P 49818201 Ki = 5.754 nM T55959 CFX2Q0 49818202 Ki = 79.43 nM T55959 C23PXY 49818203 Ki = 5.012 nM T55959 CR40BA 49836386 IC50 = 6900 nM T55959 C0M5XC 49836496 IC50 = 2100 nM T55959 CX9M3E 49837912 Ki > 10000 nM T55959 CZJV13 49852019 IC50 = 7.3 nM T55959 CSL8M9 49852020 IC50 = 2.3 nM T55959 CWCY74 49852021 IC50 = 1.5 nM T55959 CI08OL 49852022 IC50 = 15 nM T55959 C1BH4A 49852023 IC50 = 3 nM T55959 COR7M1 49863727 Ki = 9.5 nM T55959 C7CJ5W 49863728 Ki = 0.6 nM T55959 C9YS5V 49863729 Ki = 0.4 nM T55959 CO3K6A 49863748 Ki = 0.5 nM T55959 CK92TE 49863749 IC50 = 2.4 nM T55959 CFZ39O 49865822 Ki = 6.31 nM T55959 CT34HY 49865823 Ki = 50.12 nM T55959 CK7O1S 49865875 Ki = 6.31 nM T55959 CCH8T4 49865876 Ki = 3.162 nM T55959 C8V3NG 49865877 Ki = 3.162 nM T55959 CEK89Q 49865878 Ki = 12.59 nM T55959 CZA5X4 49865879 Ki = 6.31 nM T55959 CD4LO5 49865880 Ki = 3.162 nM T55959 CZ2W8K 49865881 Ki = 794.33 nM T55959 C0R8AN 49865934 Ki = 39.81 nM T55959 C9TN8D 49865935 Ki = 63.1 nM T55959 C3YJ4G 49865936 Ki = 2.512 nM T55959 CB5WR8 49865937 Ki = 3.981 nM T55959 C8LJ4H 49865983 Ki = 1.259 nM T55959 C1MPT6 49865984 Ki = 2.512 nM T55959 C62NWE 49865985 Ki = 3.981 nM T55959 C5H4AY 49865986 Ki = 1 nM T55959 C90XRC 49865987 Ki = 1.995 nM T55959 CKMX26 49866033 IC50 = 78 nM T55959 CEFJ14 49866038 Ki = 10 nM T55959 CZ9I3O 49866039 Ki = 3.162 nM T55959 C96XFK 49866040 Ki = 63.1 nM T55959 C26NLJ 49866041 Ki = 7.943 nM T55959 CQHM34 49866042 Ki = 1 nM T55959 CK1Y3B 49866085 IC50 = 91.7 nM T55959 C8JY3K 49866095 Ki = 12.59 nM T55959 C9N5CZ 49866096 Ki = 10 nM T55959 CC1L4U 49866097 Ki = 15.85 nM T55959 CV49QI 49866161 Ki = 5.012 nM T55959 CF59UG 49866162 Ki = 79.43 nM T55959 C5N8KG 49866163 Ki = 3.981 nM T55959 C4F8UX 49866191 Ki = 7.943 nM T55959 C2RY0J 50878551 Ki = 3162.28 nM T55959 C1W6TV 50898777 Ki > 10000 nM T55959 CXMZ73 50898778 Ki > 10000 nM T55959 C2CYL1 50917604 Ki = 86.7 nM T55959 C0C9HA 50917605 Ki = 5.6 nM T55959 C9U6BI 50917780 Ki = 106 nM T55959 C6JNK5 50917781 Ki = 17.9 nM T55959 C1C9JT 50917784 Ki = 127 nM T55959 C1BMO5 50917785 Ki = 4.1 nM T55959 C8J5MB 50941458 IC50 = 5033 nM T55959 CJP82R 50941459 IC50 = 246 nM T55959 CJ43IF 50941460 IC50 = 39 nM T55959 CIGJ83 50942207 IC50 = 7 nM T55959 CK4HM2 50942208 IC50 = 7.2 nM T55959 C2SHO8 50993865 IC50 = 72 nM T55959 CX48AD 51002362 Ki = 3221 nM T55959 C6LVM3 51003382 Ki > 6460 nM T55959 CIW56N 51003383 Ki > 6460 nM T55959 CE4KP1 51050257 Ki > 10000 nM T55959 CYR7P8 51346818 IC50 = 21 nM T55959 CD4B6S 51346820 IC50 = 90 nM T55959 CV8P2U 51353528 IC50 = 2800 nM T55959 CANW89 52943609 IC50 = 11 nM T55959 CJV4D0 52946564 IC50 = 4000 nM T55959 CYX21V 52948756 Ki = 77 nM T55959 C8XB1M 52949040 IC50 = 6600 nM T55959 COB3C8 52949721 Ki = 6.3 nM T55959 C42NYA 53248999 Ki = 63.1 nM T55959 C6HKP5 53316563 Ki = 2056 nM T55959 CKS81C 53316705 IC50 = 65 nM T55959 CVZ7U8 53316706 IC50 = 32.7 nM T55959 CB01DE 53316707 IC50 = 46.6 nM T55959 C6IHN7 53316708 IC50 = 157 nM T55959 CGQJ07 53316788 Ki > 6460 nM T55959 CR41UN 53316822 IC50 = 454 nM T55959 CL78NK 53316823 IC50 = 103 nM T55959 CB86XC 53316913 IC50 = 1318 nM T55959 CE26AQ 53317143 IC50 = 1 nM T55959 C2V6WS 53317144 IC50 < 1 nM T55959 C9L6YK 53317145 IC50 = 9 nM T55959 CST69D 53317146 IC50 = 42 nM T55959 CS9Z0R 53317167 IC50 = 884 nM T55959 CH76LD 53317168 IC50 = 11 nM T55959 C63XCS 53317410 IC50 = 173 nM T55959 C9RNL2 53317411 IC50 > 10000 nM T55959 CPK1R2 53317591 IC50 = 155 nM T55959 CU2R4V 53317717 IC50 > 1000 nM T55959 CZTW58 53317736 Ki = 2040 nM T55959 CIK7D3 53317746 IC50 = 22 nM T55959 CW0G5B 53318001 IC50 = 139 nM T55959 C7APQ5 53318002 IC50 = 69.2 nM T55959 CRHA45 53318003 IC50 > 2000 nM T55959 C1HO3W 53318004 IC50 = 126 nM T55959 C68GHK 53318005 IC50 = 238 nM T55959 CW70NZ 53318092 Ki = 2190 nM T55959 C7PC1G 53318093 Ki > 3880 nM T55959 CQ37BK 53318094 Ki = 2030 nM T55959 C8RLQ9 53318095 Ki > 5870 nM T55959 C85UKZ 53318218 IC50 = 737 nM T55959 CFHE24 53318434 IC50 < 1 nM T55959 CI49RQ 53318452 IC50 = 3639 nM T55959 CWHC74 53318453 IC50 = 625 nM T55959 CD0Y4B 53318705 IC50 > 10000 nM T55959 CE1W5G 53318706 IC50 > 10000 nM T55959 C8C7YZ 53318707 IC50 = 481 nM T55959 C8PAY5 53318980 IC50 = 1777 nM T55959 CZ0M8J 53319021 IC50 = 91 nM T55959 C8V1AW 53319232 IC50 = 465 nM T55959 C7BY4O 53319345 IC50 = 456 nM T55959 C5FRP2 53319428 Ki > 4860 nM T55959 CY65NV 53319429 Ki > 5940 nM T55959 C1MD0J 53319430 Ki = 312 nM T55959 C1E7BF 53319431 Ki > 5590 nM T55959 C2OJW5 53319432 Ki > 5870 nM T55959 CT0W3X 53319433 Ki > 4620 nM T55959 C8EKT2 53319478 IC50 = 273 nM T55959 C79JCL 53319479 IC50 = 11 nM T55959 CK2G3D 53319480 IC50 = 111 nM T55959 CVXT03 53319481 IC50 = 484 nM T55959 C90TZS 53319482 IC50 = 212 nM T55959 CJH1M0 53319767 IC50 = 2 nM T55959 CZ6L5C 53319784 IC50 = 83 nM T55959 CE6V4A 53319785 IC50 = 739 nM T55959 C63JGV 53319832 IC50 = 63 nM T55959 CVF5U0 53319835 IC50 = 268 nM T55959 CXF1S4 53320328 IC50 = 125 nM T55959 C6RB3C 53320515 Ki = 517 nM T55959 CODA90 53320569 Ki = 3443 nM T55959 CZE80U 53320651 IC50 = 12 nM T55959 CQC23J 53320652 IC50 = 14 nM T55959 C19ZWJ 53320686 IC50 = 605 nM T55959 CB84NG 53320778 IC50 = 62 nM T55959 C8JX4C 53320779 IC50 = 45 nM T55959 CP7RZ3 53320780 IC50 = 92 nM T55959 CL67KH 53320781 IC50 = 339 nM T55959 CK5C0S 53320864 IC50 = 380 nM T55959 CQ90IR 53321058 IC50 = 1 nM T55959 CZ7NM6 53321059 IC50 = 395 nM T55959 CXY92R 53321081 IC50 = 57 nM T55959 CS42VL 53321082 IC50 = 546 nM T55959 CO7L6Z 53321083 IC50 = 3 nM T55959 CSY1K4 53321125 IC50 = 9 nM T55959 CAJ4L7 53321331 IC50 > 10000 nM T55959 CMZ7F8 53321332 IC50 = 8066 nM T55959 CZEF75 53321509 IC50 = 332 nM T55959 C1AI0C 53321510 IC50 = 130 nM T55959 CSX14G 53321869 Ki = 1.2 nM T55959 C34ORB 53321945 IC50 > 2000 nM T55959 C6ND9H 53321946 IC50 = 49 nM T55959 C4X3IS 53321979 IC50 = 12 nM T55959 CLQ85U 53322027 Ki > 6370 nM T55959 C53HJK 53322028 Ki > 6460 nM T55959 CLD82J 53322084 IC50 = 114 nM T55959 C7QF2E 53322085 IC50 = 319 nM T55959 CY09UA 53322086 IC50 = 559 nM T55959 CBUT35 53322087 IC50 = 1616 nM T55959 CXL8W9 53322200 IC50 = 2427 nM T55959 CE63PO 53322201 IC50 = 2775 nM T55959 C3M9SC 53322397 IC50 = 4 nM T55959 CLT3Q2 53322398 IC50 = 2 nM T55959 CZLT60 53322409 IC50 = 17 nM T55959 CLZ41J 53322410 IC50 = 384 nM T55959 C3YWZ5 53322451 IC50 = 36 nM T55959 CZ92BF 53322452 IC50 = 350 nM T55959 C5G8RQ 53322642 IC50 > 10000 nM T55959 CV49EH 53322836 IC50 = 43.5 nM T55959 CRUF31 53322954 Ki > 6220 nM T55959 C6UBF1 53323137 Ki = 4.5 nM T55959 CNCG12 53323138 Ki = 363 nM T55959 C0CSA9 53323139 Ki = 2754 nM T55959 C9U1CI 53323140 Ki = 658 nM T55959 C3HKJ0 53323299 IC50 > 5000 nM T55959 C6ZFR5 53323300 IC50 = 101.3 nM T55959 CK6U0Y 53323301 IC50 = 497 nM T55959 CGA5R8 53323302 IC50 = 269 nM T55959 CND26W 53323338 IC50 = 122 nM T55959 C6KAN9 53323339 IC50 = 309 nM T55959 C2OB7G 53323389 Ki > 6410 nM T55959 C4UBX5 53323390 Ki > 6410 nM T55959 C1WU4E 53323391 Ki = 4510 nM T55959 CGN6Z3 53323531 IC50 > 10000 nM T55959 CAQ07J 53323532 IC50 = 201 nM T55959 C1GZ3B 53323533 IC50 = 1404 nM T55959 C4D1LX 53323761 IC50 = 12 nM T55959 CPKM07 53323762 IC50 = 2 nM T55959 CQW2S7 53323771 IC50 = 1 nM T55959 CO7TC1 53323812 IC50 = 1520 nM T55959 CDRV76 53323814 IC50 = 30 nM T55959 C32YWL 53324045 Ki = 121 nM T55959 C98OKX 53324333 IC50 = 125 nM T55959 C46XAC 53324366 IC50 = 177 nM T55959 C36USG 53324493 Ki = 1112 nM T55959 CR4W9L 53324553 Ki = 1684 nM T55959 CCK4T2 53324628 IC50 = 66.5 nM T55959 CW58QL 53324656 IC50 = 100 nM T55959 CFJ1B0 53324709 Ki > 4260 nM T55959 C5I1FG 53324762 IC50 = 176 nM T55959 C94GOI 53324763 IC50 = 111 nM T55959 COP3J6 53324764 IC50 = 332 nM T55959 CE7DZ0 53324844 IC50 = 2261 nM T55959 CB34ZM 53325028 IC50 = 82 nM T55959 CY9H2U 53325042 IC50 = 170 nM T55959 CRQF15 53325242 Ki = 529 nM T55959 C3QNR2 53325463 IC50 = 8 nM T55959 CAGT23 53325525 IC50 > 1000 nM T55959 CZN8B4 53325581 IC50 = 281 nM T55959 COZ1W9 53325647 IC50 = 2010 nM T55959 CB37XF 53325861 Ki = 101 nM T55959 C1N7XO 53325966 IC50 = 16 nM T55959 CZ69OW 53326010 Ki = 2090 nM T55959 CZ1U9T 53326011 Ki = 4700 nM T55959 CM7YA0 53326118 IC50 = 804 nM T55959 CJ6G7X 53326119 IC50 = 750 nM T55959 CTH12B 53326554 IC50 = 8710 nM T55959 CG24AT 53381002 IC50 > 10000 nM T55959 C0M5WU 53391513 IC50 = 3388.44 nM T55959 C8DR9L 53391514 IC50 = 1000 nM T55959 C7GH1I 53391515 IC50 = 9772.37 nM T55959 C3BX4K 53391516 IC50 = 3311.31 nM T55959 C5B1ST 53391517 IC50 = 20.42 nM T55959 CQYB97 53391614 IC50 = 2818.38 nM T55959 CK3D9F 53391615 IC50 > 10000 nM T55959 C3S5QX 53391616 IC50 > 10000 nM T55959 CI3T5Y 53391617 IC50 = 9772.37 nM T55959 CKOD62 53391618 IC50 = 100 nM T55959 CD24UN 53391714 IC50 = 28.84 nM T55959 CA0GN6 53391715 IC50 = 2454.71 nM T55959 CQ4E2W 53391716 IC50 = 61.66 nM T55959 C64TJO 53391717 IC50 = 33.88 nM T55959 C3Q6IL 53391718 IC50 = 30.2 nM T55959 C7UBN1 53392848 IC50 = 1023.29 nM T55959 CB5JU8 53392849 IC50 = 489.78 nM T55959 C0JI1M 53392850 IC50 = 478.63 nM T55959 CPIT32 53392851 IC50 = 501.19 nM T55959 C8K1TZ 53392852 IC50 = 158.49 nM T55959 CS7TE6 53392939 IC50 = 1288.25 nM T55959 CT7U5L 53392940 IC50 = 416.87 nM T55959 COES13 53466370 IC50 = 870 nM T55959 CMOZ61 53475319 Ki = 205 nM T55959 CDV82B 53492877 IC50 = 2190 nM T55959 C9ZUX3 53667258 IC50 = 2143 nM T55959 CNV45T 54345800 IC50 = 32.7 nM T55959 CREO89 54377055 IC50 = 22.7 nM T55959 CHE5Q4 54380151 Ki = 290 nM T55959 CEY2B8 54583277 IC50 = 44 nM T55959 C6ME0B 54584239 IC50 = 61 nM T55959 CL5I1R 54753271 Ki = 5000 nM T55959 CGO9V3 54756922 IC50 = 1035 nM T55959 CYS19X 54756924 IC50 = 964 nM T55959 CLC71N 54756925 IC50 = 479 nM T55959 CF82MX 54756926 IC50 = 341 nM T55959 CY7IR2 54757020 IC50 = 792 nM T55959 COJ0T5 54757025 IC50 = 599 nM T55959 CGT6F0 54757120 IC50 = 211 nM T55959 C4S6UM 54757121 IC50 = 2040 nM T55959 CB87MF 54766009 IC50 = 356.6 nM T55959 CLV3N6 54767240 IC50 = 247.2 nM T55959 CZ47UJ 54767241 IC50 = 238.1 nM T55959 C5RX1P 54767242 IC50 = 602.1 nM T55959 C32NWX 54767413 IC50 = 986.1 nM T55959 C6ASW2 54767576 IC50 = 863.1 nM T55959 CO6CJ2 54767906 IC50 = 8192.5 nM T55959 CMJ32F 56659126 Ki = 31.62 nM T55959 CQ6XM7 56659146 Ki = 25.12 nM T55959 CFT9V8 56659147 Ki = 15.85 nM T55959 CO0GR7 56659199 Ki = 0.1585 nM T55959 CC26HR 56659200 Ki = 63.1 nM T55959 CGID30 56659201 Ki = 3.162 nM T55959 CG0M7T 56662629 Ki = 6.31 nM T55959 CP2ZS4 56662647 Ki = 19.95 nM T55959 C8NIZ3 56662648 Ki = 3.981 nM T55959 CN7WB5 56662696 Ki = 15.85 nM T55959 CD9F3J 56662697 Ki = 25.12 nM T55959 CH37LU 56663451 IC50 > 10000 nM T55959 C5HF9D 56666091 Ki = 19.95 nM T55959 C9RE3V 56669493 Ki = 15.85 nM T55959 CK3R7P 56669494 Ki = 199.53 nM T55959 CVRH79 56669561 Ki = 6.31 nM T55959 CC9XR7 56669562 Ki = 15.85 nM T55959 CXE9A8 56669563 Ki = 3.162 nM T55959 CNK39V 56673078 Ki = 1 nM T55959 C93KBW 56679646 Ki = 1.259 nM T55959 CAR8M5 56679647 Ki = 12.59 nM T55959 CN1C3K 56679724 Ki = 0.7943 nM T55959 CET3N2 56682964 Ki = 7.943 nM T55959 CK73UC 56683046 Ki = 0.1995 nM T55959 CZR91E 56683047 Ki = 1.995 nM T55959 C60IBF 56683048 Ki = 1.585 nM T55959 C90DOS 56942993 IC50 = 140 nM T55959 CHN2F6 56949640 Ki = 24 nM T55959 CZI53T 56961001 IC50 > 10000 nM T55959 C1TC7Q 56963799 Ki = 137 nM T55959 CCJ93V 57391031 Ki = 82.2 nM T55959 C8XV3D 57391453 Ki = 3071 nM T55959 CFT5U6 57391594 Ki = 501.19 nM T55959 CUR6W7 57391595 Ki = 371.54 nM T55959 CYFN26 57391657 Ki = 0.5012 nM T55959 C9LX1S 57391709 Ki = 0.87 nM T55959 CGN17Y 57391710 Ki = 9.55 nM T55959 CH2I3S 57393445 Ki = 0.6026 nM T55959 CRN9S1 57395067 Ki = 501.19 nM T55959 C45CVE 57395127 Ki = 70.79 nM T55959 C6SZ4E 57396296 Ki = 7.9 nM T55959 C6HBG0 57396813 IC50 = 6300 nM T55959 CWN71D 57396838 Ki = 501.19 nM T55959 CJ8A7B 57402008 Ki = 371.54 nM T55959 CP03KF 57403872 Ki = 89.13 nM T55959 C4N3VY 57403918 Ki = 116 nM T55959 C8J3EP 57403921 Ki = 0.3981 nM T55959 CLWD45 57459488 Ki = 5005 nM T55959 CHU5T7 57523687 EC50 = 70 nM T55959 C0WJ4E 58954830 IC50 = 13 nM T55959 CSF52J 58954867 IC50 = 41 nM T55959 C9ZP3D 58954900 IC50 = 167 nM T55959 CHQE32 58954945 IC50 = 518 nM T55959 CA36QL 59800034 IC50 = 78600 nM T55959 C3K5JN 60165681 Ki = 4742 nM T55959 C3XL7O 66561967 Ki > 10000 nM T55959 CGF3J5 66572162 IC50 = 491 nM T55959 CZL90M 66572393 IC50 = 566 nM T55959 C2UZ3A 66572397 IC50 = 564 nM T55959 CCR2I5 66572399 IC50 = 689 nM T55959 C78XLS 66813470 IC50 = 2000 nM T55959 CL8R5V 66975152 IC50 > 1000 nM T55959 C0OC8T 66975291 IC50 > 1000 nM T55959 CCN1W5 66975591 IC50 > 1000 nM T55959 C23DPF 66975638 IC50 = 70 nM T55959 C3W0XI 66975648 IC50 > 10000 nM T55959 C51JHP 66975671 IC50 = 1400 nM T55959 CV19LA 66975764 IC50 = 130 nM T55959 C50HKX 66975948 IC50 > 1000 nM T55959 C0L2QJ 66976018 IC50 > 10000 nM T55959 CE9A4J 66976134 IC50 > 1000 nM T55959 CZE5S6 66976296 IC50 = 400 nM T55959 C78MWK 66976356 IC50 > 1000 nM T55959 C5EM9P 66976389 IC50 > 1000 nM T55959 CP3M9I 66976532 IC50 = 1500 nM T55959 CAL40U 66976565 IC50 = 240 nM T55959 CI29HX 66976607 IC50 = 66 nM T55959 C6I7SV 66976613 IC50 = 3100 nM T55959 C8LD7M 66976718 IC50 > 10000 nM T55959 C6ON5Y 66976777 IC50 > 1000 nM T55959 C0MYB6 68653619 Ki = 140 nM T55959 CNY0W5 68673707 IC50 = 71 nM T55959 C76ROM 68673872 IC50 = 40 nM T55959 CD3U6K 68731121 Ki > 10000 nM T55959 CSF80C 68993720 IC50 > 300 nM T55959 CVZ51D 68993987 IC50 = 16 nM T55959 CN0MY2 68994312 IC50 = 9 nM T55959 CKTA56 68994365 IC50 = 7.5 nM T55959 CE1WF3 68994389 IC50 = 11 nM T55959 CN08VY 68994725 IC50 = 5.8 nM T55959 C0ZY9I 68994988 IC50 = 88 nM T55959 CR3H9X 68995479 IC50 = 23 nM T55959 C1LWS9 68995587 IC50 = 110 nM T55959 CDLR80 68995667 IC50 = 4.5 nM T55959 CCIV97 68995742 IC50 = 12 nM T55959 C2MK1S 68995928 IC50 = 51 nM T55959 C56VJS 68996260 IC50 = 5.7 nM T55959 CQ4Y2V 68996331 IC50 = 43 nM T55959 CHI19N 68996402 IC50 = 12 nM T55959 C17BRZ 68997664 IC50 = 6.9 nM T55959 CDT9Z5 68998740 IC50 = 890 nM T55959 CP0AR5 68999429 IC50 = 66 nM T55959 CN14QD 69000395 IC50 = 5.3 nM T55959 C6IP8Q 69082816 Ki > 10000 nM T55959 CNM1U4 69397184 Ki = 291 nM T55959 CYM94S 70676472 IC50 = 32 nM T55959 C7J0FD 70676474 IC50 = 72 nM T55959 CLTA38 70676476 IC50 = 35 nM T55959 CMN57J 70676478 IC50 = 54 nM T55959 C9QZ7C 70676480 IC50 = 148 nM T55959 C09HRL 70681048 IC50 = 102 nM T55959 CURI86 70681049 IC50 > 3000 nM T55959 CIX1V8 70681050 IC50 > 3000 nM T55959 C17ITX 70681051 IC50 = 356 nM T55959 C4ZK7S 70681052 IC50 = 64 nM T55959 CU32RF 70681053 IC50 > 1000 nM T55959 C4AVG9 70681054 IC50 > 1000 nM T55959 CU48EX 70681055 IC50 = 9 nM T55959 C7W3JA 70681326 Ki = 19.95 nM T55959 C67CHV 70681491 Ki > 10000000 nM T55959 CT65MH 70681573 Ki = 3309 nM T55959 C4YQ2E 70682258 Ki = 9.1 nM T55959 CIE30Z 70683174 IC50 > 3000 nM T55959 C7X4VF 70683175 IC50 = 139 nM T55959 CP07IW 70683176 IC50 > 1000 nM T55959 C39QGY 70683608 Ki > 10000000 nM T55959 C7HM6W 70685249 IC50 > 3000 nM T55959 CQ8Y0N 70685250 IC50 > 3000 nM T55959 CC2L8W 70685251 IC50 > 3000 nM T55959 CFQ1I9 70685252 IC50 > 1000 nM T55959 CDI70T 70685253 IC50 > 1000 nM T55959 C8FQ6K 70685254 IC50 = 1720 nM T55959 C60SBP 70685515 Ki = 199.53 nM T55959 CCOR65 70685727 Ki > 10000000 nM T55959 C3UBM6 70687401 IC50 > 3000 nM T55959 C05OPN 70687402 IC50 = 487 nM T55959 CJ9Q6Y 70687403 IC50 = 20 nM T55959 C1CH5A 70687667 Ki = 125.89 nM T55959 CTVW13 70689263 IC50 = 325 nM T55959 C7RA0K 70689264 IC50 = 207 nM T55959 CKMJ68 70689265 IC50 = 540 nM T55959 C4E3BZ 70689455 IC50 = 349 nM T55959 C3OJY2 70689456 IC50 > 1000 nM T55959 CU84XH 70689457 IC50 > 1000 nM T55959 C8NH5V 70689458 IC50 > 1000 nM T55959 CWL42U 70690666 Ki = 4 nM T55959 CB58JU 70691565 IC50 = 272 nM T55959 C3KS4O 70691566 IC50 > 3000 nM T55959 C5JPR4 70691567 IC50 = 13 nM T55959 C7R0NO 70691568 IC50 > 3000 nM T55959 CS08ZT 70691569 IC50 > 1000 nM T55959 CF63DA 70691570 IC50 > 1000 nM T55959 CP8ZB4 70691571 IC50 = 39 nM T55959 CVF95N 70691572 IC50 = 18 nM T55959 CMH98F 70691573 IC50 = 350 nM T55959 C59NVG 70691872 IC50 = 15.85 nM T55959 C4A7QI 70692139 Ki = 2309 nM T55959 CB3NW6 70693452 IC50 = 430 nM T55959 CP38FE 70693453 IC50 = 1.35 nM T55959 C7RF8K 70693651 IC50 > 3000 nM T55959 C6R4EB 70693652 IC50 = 336 nM T55959 CP5I2J 70693653 IC50 > 3000 nM T55959 CYS1E6 70693654 IC50 > 3000 nM T55959 CR30AX 70693655 IC50 > 3000 nM T55959 C8LP2J 70693656 IC50 > 40000 nM T55959 C8IQC6 70695563 IC50 = 25 nM T55959 C5DP3J 70695564 IC50 = 15.7 nM T55959 CRXH46 70695767 IC50 > 10000 nM T55959 CJ01ST 70695768 IC50 > 10000 nM T55959 C25SJC 70695769 IC50 > 3000 nM T55959 CRS3M8 70695770 IC50 = 110 nM T55959 CFM5Z8 70695771 IC50 = 370 nM T55959 CN9RQ3 70695772 IC50 > 1000 nM T55959 C7P9IB 70696895 Ki = 35 nM T55959 C37USC 70697274 Ki = 10.6 nM T55959 CB9H4S 70697574 IC50 = 238 nM T55959 CI93FE 70963695 IC50 > 10000 nM T55959 C2FN8M 71134973 IC50 > 1000 nM T55959 C5BER9 71332336 IC50 = 10000 nM T55959 C5X3LM 71450608 Ki = 1840 nM T55959 C87FQH 71450609 Ki = 687 nM T55959 C68BJU 71450818 IC50 = 12 nM T55959 C4TWS5 71452172 Ki = 373 nM T55959 CIC65E 71454201 Ki = 8 nM T55959 CFBC49 71455896 Ki > 10000 nM T55959 CCY4E2 71456314 IC50 = 19 nM T55959 C7MNB5 71457264 Ki = 2899 nM T55959 C6X1GN 71457767 Ki = 36.2 nM T55959 C87FDI 71458022 Ki = 510 nM T55959 CP16SV 71458086 IC50 = 14.1 nM T55959 CK5T4P 71459604 Ki = 3180 nM T55959 C3L2SU 71461395 Ki > 8500 nM T55959 CX69JF 71461719 IC50 = 14.2 nM T55959 CKX5O8 71463061 Ki > 10000 nM T55959 CD3L7R 71463125 Ki = 210 nM T55959 C4RAQ6 71518063 Ki = 10900 nM T55959 CO26TC 71541094 Ki = 8 nM T55959 CE8YO0 71541095 Ki = 11 nM T55959 CN79ZY 71541096 Ki = 37 nM T55959 CNCR14 71541097 Ki = 9 nM T55959 CW34SU 71541098 Ki = 5 nM T55959 CKW24J 71541099 Ki = 3 nM T55959 C0ZL6O 71541186 Ki = 13 nM T55959 C92PZK 71541187 Ki = 23 nM T55959 C0T4RD 71541188 Ki = 60 nM T55959 CB91FO 71541189 Ki = 6 nM T55959 CY5E0J 71541190 Ki = 6 nM T55959 C4XK1S 71541191 Ki = 8 nM T55959 C32HNI 71541192 Ki = 10 nM T55959 C9C0JU 71541193 Ki = 49 nM T55959 CFO05K 71541194 Ki = 24 nM T55959 CD1T5J 71541195 Ki = 68 nM T55959 CBWZ86 71541287 Ki = 25 nM T55959 CK82YE 71541288 Ki = 240 nM T55959 CQ81HF 71541289 Ki = 23 nM T55959 CU53JE 71541292 Ki = 6 nM T55959 C57KER 71541293 Ki = 400 nM T55959 C4A7KU 71550921 EC50 = 2700 nM T55959 C6B3CF 71562265 Ki = 1000 nM T55959 C9V0FZ 71562266 Ki = 1000 nM T55959 C49VSK 71562370 Ki = 251.19 nM T55959 COFY97 71562371 Ki = 158.49 nM T55959 C1JCZ5 71562372 Ki = 125.89 nM T55959 CXR0E7 71562373 Ki = 63.1 nM T55959 C4PDM8 71562374 Ki = 50.12 nM T55959 C3L9HK 71562375 Ki = 125.89 nM T55959 CX7VK3 71562376 Ki = 31.62 nM T55959 CHW7K1 71562377 Ki = 15.85 nM T55959 CK95GV 71562472 Ki = 158.49 nM T55959 C4NS5W 71562473 Ki = 125.89 nM T55959 CH49FE 71562477 Ki = 39.81 nM T55959 CU1CZ6 71562478 Ki = 3.162 nM T55959 CPAY18 71562479 Ki = 39.81 nM T55959 CY39RM 71562586 Ki = 125.89 nM T55959 C4F2UW 71562587 Ki = 316.23 nM T55959 CI3KA2 71562588 Ki = 316.23 nM T55959 C13NIO 71562589 Ki = 63.1 nM T55959 CKPH80 71562590 Ki = 100 nM T55959 C0NIA6 71562591 Ki = 100 nM T55959 CRCT65 71562592 Ki = 398.11 nM T55959 C1XQ5M 71562593 Ki = 125.89 nM T55959 CFQP86 71562712 Ki = 2511.89 nM T55959 CPDV40 71562713 Ki = 39.81 nM T55959 CP2N3Y 71562714 Ki = 794.33 nM T55959 CS59VG 71562715 Ki = 398.11 nM T55959 CE7X9R 71562716 Ki = 100 nM T55959 CP20LV 71562717 Ki = 100 nM T55959 CQU78X 71562718 Ki = 125.89 nM T55959 CCO48Y 71562719 Ki = 316.23 nM T55959 CSYR25 71562833 Ki = 12.59 nM T55959 CF0R4S 71562834 Ki = 63.1 nM T55959 C5NO2C 71562835 Ki = 63.1 nM T55959 C2UQD4 71562836 Ki = 100 nM T55959 C1Q4JZ 71562837 Ki = 79.43 nM T55959 CNQ2J1 71575525 Ki = 1800 nM T55959 CJPR13 71625847 IC50 = 290 nM T55959 CZWN24 71716486 Ki = 100 nM T55959 CH8O3Z 71717705 Ki = 100 nM T55959 C0O4ID 71718185 Ki = 4.2 nM T55959 C7TCH6 71718282 Ki = 62 nM T55959 CF2AW7 71719112 IC50 = 482 nM T55959 CM7T0H 71719533 Ki = 7.943 nM T55959 C2EWG5 71719830 Ki = 91 nM T55959 CY6DR8 71727648 IC50 = 160 nM T55959 CA3H0X 71727754 IC50 = 2400 nM T55959 C2WD4V 71727756 IC50 = 170 nM T55959 CDT2P5 71727758 IC50 = 79 nM T55959 C39EUA 71727760 IC50 = 72 nM T55959 C8BLG9 71727762 IC50 = 2200 nM T55959 C1XB7U 71727764 IC50 = 220 nM T55959 CS83FB 71727766 IC50 = 97 nM T55959 CX7O8K 71727768 IC50 = 190 nM T55959 CEM15Z 71727886 IC50 = 180 nM T55959 C5BL4F 71727888 IC50 = 100 nM T55959 CX21QS 71727890 IC50 = 26 nM T55959 COUT12 71812204 IC50 = 180 nM T55959 CT03WY 72202713 IC50 = 36.6 nM T55959 CKS1Z3 72202714 IC50 = 8.14 nM T55959 CJM9I7 72202715 IC50 = 17.3 nM T55959 CIR13D 72202716 IC50 = 36.3 nM T55959 C91REH 72202846 IC50 = 38.7 nM T55959 CTL7Z6 72202847 IC50 = 1731 nM T55959 C1UO9J 72202848 IC50 = 33.1 nM T55959 CJ7VK8 72202849 IC50 = 171.9 nM T55959 C4V2NE 72202850 IC50 = 280.6 nM T55959 CDG0A8 72202852 IC50 = 159.7 nM T55959 CV5TJ6 72202983 IC50 = 120.9 nM T55959 C3ZHJ1 72202984 IC50 = 284.7 nM T55959 CWH6T3 72548703 IC50 = 4.9 nM T55959 C48RGH 72737188 Ki = 36.99 nM T55959 CAEQ04 72737189 Ki = 1.33 nM T55959 CC65OA 73213195 Ki > 10000 nM T55959 CW83DK 73213196 Ki > 10000 nM T55959 C0HTU4 73345764 IC50 = 10.9 nM T55959 CRG9J8 73346332 Ki = 4523 nM T55959 CK0HR9 73346334 Ki = 2016 nM T55959 CK48PN 73347369 Ki > 890 nM T55959 C4YV6S 73347524 IC50 = 500 nM T55959 CEQS50 73347526 IC50 = 1700 nM T55959 CI0JV6 73347528 IC50 = 580 nM T55959 CY60RD 73347826 Ki = 1558 nM T55959 CFW96K 73347828 Ki > 10000 nM T55959 C85LKM 73348886 Ki = 354 nM T55959 C9Y6OD 73348887 Ki > 890 nM T55959 CM50LN 73349057 IC50 = 1100 nM T55959 C7XOF4 73349320 IC50 = 99.6 nM T55959 CQH3J5 73349358 Ki > 10000 nM T55959 CHNT68 73350623 IC50 = 470 nM T55959 C87LGB 73352415 Ki = 1293 nM T55959 CCD70L 73353582 IC50 = 2600 nM T55959 CYPL06 73355375 IC50 = 41.7 nM T55959 C4F7VK 73355415 Ki = 126 nM T55959 CAI63V 73355417 Ki = 3480 nM T55959 C10ASZ 73355420 Ki > 10000 nM T55959 CWK70C 73356510 Ki > 890 nM T55959 C2E7QW 75201901 Ki = 8300 nM T55959 CRK8G2 76314641 Ki = 2300 nM T55959 C4G6RW 76335160 Ki = 12.5 nM T55959 C28RIZ 76518514 Ki = 778 nM T55959 C2U0BG 87055263 IC50 = 390 nM T55959 C2LQ5Z 89437491 IC50 = 362.8 nM T55959 C2BM9L 89768534 IC50 = 175 nM T55959 CB4Y7R 89768546 IC50 = 150 nM T55959 CP29UR 89838714 IC50 > 1000 nM T55959 CF6P3I 89843681 IC50 > 1000 nM T55959 CT8HK6 90389439 Ki = 101 nM T55959 CU9ED1 90389592 Ki = 1200 nM T55959 CBH87U 91667621 IC50 = 38 nM T55959 C0RV4M 91799659 IC50 = 160 nM T55959 CCY0O2 100951644 IC50 = 61000 nM T55959 C5E3PB 101882704 Ki = 557 nM T55959 C10DAF 112777136 IC50 = 91380 nM T55959 CI3KM2 118103909 IC50 = 2870 nM T55959 CAIU03 118104096 IC50 = 3290 nM T55959 C7AYV5 118540795 Ki = 2120 nM T55959 C2I0HB 118643968 Ki = 6.5 nM T55959 CF5K0V 118691439 Ki > 9300 nM T55959 CW15HU 118700678 Ki > 7100 nM T55959 CA79GZ 118706038 IC50 = 53.6 nM T55959 CGBC58 118706039 IC50 = 52.1 nM T55959 C5LCJ1 118706532 IC50 = 129 nM T55959 CI2FN5 118706536 IC50 = 33.1 nM T55959 C2BG1F 118706537 IC50 = 82.5 nM T55959 C2WP6X 118706538 IC50 = 63.9 nM T55959 CZE4U0 118706539 IC50 = 35.6 nM T55959 CX8I0G 118706540 IC50 = 143 nM T55959 C4S9VT 118706541 IC50 = 164 nM T55959 CKD94F 118706542 IC50 = 162 nM T55959 C0KQO9 118706543 IC50 = 80.4 nM T55959 C5HJY0 118706544 IC50 = 110 nM T55959 CJ15AS 118708361 IC50 = 420 nM T55959 C7XEC0 118708362 IC50 = 4000 nM T55959 CK30WF 118708364 IC50 = 8100 nM T55959 CG7W4D 118708365 IC50 = 4500 nM T55959 C6UJC5 118708366 IC50 > 10000 nM T55959 CLQ52I 118708373 IC50 > 10000 nM T55959 CSB25E 118709750 Ki = 285 nM T55959 CD4S9R 118709751 Ki = 354 nM T55959 CD34IY 118710582 IC50 = 3.1 nM T55959 CD1O7G 118710583 IC50 = 1400 nM T55959 C5GRY0 118713756 IC50 = 498 nM T55959 C4VAE0 118713757 IC50 = 678 nM T55959 CPDB78 118713768 IC50 = 696 nM T55959 C84GOU 118713773 IC50 = 265 nM T55959 CW0SN9 118713774 IC50 = 684 nM T55959 CUN71K 118713775 IC50 = 540 nM T55959 C6ZL1K 118713793 IC50 = 150 nM T55959 CQFH60 118713795 IC50 = 187 nM T55959 CC58ZS 118713797 IC50 = 327 nM T55959 C2LY9D 118713799 IC50 = 118 nM T55959 CMO2V7 118713801 IC50 = 330 nM T55959 C9LKI0 118713803 IC50 = 533 nM T55959 CD2C1A 118713804 IC50 = 406 nM T55959 C2OZ7H 118713805 IC50 = 415 nM T55959 CM4P8X 118713806 IC50 = 394 nM T55959 C7EXQ9 118713807 IC50 = 441 nM T55959 C05FSJ 118714012 IC50 = 325.4 nM T55959 CVH14M 118714014 IC50 = 852.3 nM T55959 C15FVH 118714017 IC50 = 291.4 nM T55959 CGC5J6 118719847 IC50 = 120 nM T55959 C6HV3B 118730351 EC50 = 35.1 nM T55959 C3LZM9 118730352 EC50 = 9.1 nM T55959 C4G3YC 118734875 Ki = 10200 nM T55959 C9AIE1 118734876 Ki = 6600 nM T55959 C5RNW2 118857804 Ki = 4170 nM T55959 C0GQF1 118857828 Ki = 1610 nM T55959 C6UHM8 118857829 Ki = 7300 nM T55959 CA03SM 118857831 Ki > 10000 nM T55959 C0FCX2 118857833 Ki > 10000 nM T55959 CU1Z8O 118857834 Ki > 10000 nM T55959 CX2RY8 118857835 Ki > 10000 nM T55959 C2ZD0T 118857837 Ki > 10000 nM T55959 CB54AQ 118857838 Ki > 10000 nM T55959 C10VOM 118871447 IC50 = 68060 nM T55959 CS7HB2 118871454 IC50 = 14730 nM T55959 CS9VI7 118871455 IC50 = 4610 nM T55959 CDU18K 118871456 IC50 = 4100 nM T55959 C1Z4TP 118871458 IC50 = 24320 nM T55959 CDO6E7 118871463 IC50 = 44060 nM T55959 C8P3BV 118871470 IC50 = 6660 nM T55959 CQ8H1J 118871471 IC50 = 3250 nM T55959 C6YC2G 118871476 IC50 = 87060 nM T55959 CK7D6O 118879529 IC50 = 8500 nM T55959 CSC5J4 121488665 Ki = 74.3 nM T55959 CUK9E2 122181877 IC50 > 1000 nM T55959 CHKY46 122181879 IC50 > 1000 nM T55959 C9TDA7 122188500 IC50 = 1350 nM T55959 CARF60 122188503 IC50 > 10000 nM T55959 C1CJQ0 122188571 EC50 > 1000 nM T55959 CJ6G5D 122188774 IC50 = 190 nM T55959 CNT50I 122188775 IC50 = 630 nM T55959 C7ODW3 122195524 Ki < 300 nM T55959 CPO7N5 124125214 IC50 = 2170 nM T55959 CLG67Z 126641948 IC50 = 300 nM T55959 CM57GR 126720252 Ki = 1070 nM T55959 CTBN56 127026052 Ki = 1995.26 nM T55959 CEJ3R5 127029340 IC50 = 21 nM T55959 CQ0ZT9 127035062 Ki = 498 nM T55959 CU49VE 127036186 Ki = 3162.28 nM T55959 CG06BD 127036932 Ki = 794.33 nM T55959 CVW71O 127036953 Ki = 2511.89 nM T55959 CWJ59Z 127051882 IC50 > 1000 nM T55959 C50GOC 130442480 Ki > 10000 nM T55959 CM04RF 130442572 Ki = 9100 nM T55959 C1RI8Q 132060720 Ki = 2163 nM T55959 CGHO19 132060770 Ki = 2959 nM T55959 CFXL21 132060812 Ki = 1555 nM T55959 CXV95T 132578504 IC50 = 1040 nM T55959 C8NUR9 132578505 IC50 = 1200 nM T55959 CGW0I7 132578506 IC50 = 1140 nM T55959 CI4OC9 132578507 IC50 = 1010 nM T55959 C5GEB2 132578508 IC50 = 820 nM T55959 C3ONX2 132578509 IC50 = 4740 nM T55959 CAVB41 132584404 Ki > 10000 nM T55959 C68AXD 134141831 Ki = 4800 nM T55959 CBU81N 134149168 Ki = 2182 nM T55959 C1GY2T 135156251 EC50 > 10000 nM T55959 C7QAS6 135873861 Ki = 293 nM T55959 C27HTA 136236310 Ki > 10000 nM T55959 CDY5T0 136236313 Ki > 10000 nM T55959 CI6R9B 136236316 Ki = 1200 nM T55959 C3QOP1 136340699 IC50 > 1000 nM T55959 C4UON5 136389176 IC50 > 1000 nM T55959 CG05IL 136389183 IC50 > 1000 nM T55959 CP0E8J 136389204 IC50 > 1000 nM T55959 CGS61F 137553161 Ki = 4750 nM T55959 CF3ZY7 137631557 IC50 = 38100 nM T55959 C5XL1N 137631893 Ki = 11 nM T55959 C1QFO5 137632421 IC50 = 5800 nM T55959 C14RKA 137632704 IC50 = 4000 nM T55959 C0C6ZL 137632750 IC50 = 1980 nM T55959 C7C6JS 137633195 IC50 = 7200 nM T55959 CCP46O 137633241 IC50 = 3000 nM T55959 CI69VT 137633306 EC50 = 1200 nM T55959 C5G0XW 137633601 EC50 = 35 nM T55959 C5GP0H 137633918 IC50 = 38600 nM T55959 C2LJW0 137634948 IC50 > 10000 nM T55959 CP07AG 137635043 IC50 = 450 nM T55959 CTFS37 137635082 Ki = 221 nM T55959 CR74SC 137635327 IC50 = 1636 nM T55959 CW9X5R 137635426 IC50 = 2231 nM T55959 CX17BR 137635648 IC50 = 4020 nM T55959 CGOI28 137636189 Ki = 10 nM T55959 C42HCS 137636472 IC50 = 3000 nM T55959 CKQ92P 137636703 IC50 = 3290 nM T55959 COH18X 137637663 IC50 = 2000 nM T55959 CL56ZQ 137637671 IC50 = 5600 nM T55959 CYOE78 137638172 IC50 = 40400 nM T55959 CD31YG 137638231 IC50 = 6000 nM T55959 C1EU5S 137638283 IC50 > 10000 nM T55959 CJI0K6 137638828 IC50 = 163 nM T55959 CBK0I8 137639266 EC50 = 53.5 nM T55959 CI5Q2P 137639497 EC50 > 1000 nM T55959 C4BXH9 137640164 IC50 = 90500 nM T55959 CV20BW 137640543 IC50 = 6810 nM T55959 CVC6R8 137640624 IC50 = 94 nM T55959 C1X0QZ 137640906 IC50 = 8320 nM T55959 C6LXC9 137640928 IC50 = 2400 nM T55959 C06KGS 137641034 IC50 = 14600 nM T55959 CWV3C4 137641359 IC50 = 56700 nM T55959 CE8N4S 137641762 EC50 > 1000 nM T55959 C9VR5M 137643839 IC50 = 2749 nM T55959 CASM14 137643954 IC50 = 29300 nM T55959 C6FPZ5 137644016 Ki = 16 nM T55959 C3ZRY2 137645338 IC50 = 3740 nM T55959 COES67 137645514 EC50 > 1000 nM T55959 C85OYG 137645602 IC50 = 97.5 nM T55959 C0JV5S 137645725 IC50 = 155700 nM T55959 C1KT5F 137645761 IC50 > 10000 nM T55959 CPZ3E1 137646230 IC50 = 608 nM T55959 CE6NB3 137646374 IC50 = 107600 nM T55959 CT7UG4 137646579 IC50 = 69100 nM T55959 C19CXJ 137647807 Ki = 147 nM T55959 CE9M3Z 137648195 IC50 = 10000 nM T55959 CIH3O8 137648265 IC50 = 679.8 nM T55959 C0EVB7 137648614 IC50 = 3640 nM T55959 CG1ME5 137648669 IC50 = 6550 nM T55959 CO4VY9 137649584 IC50 = 4900 nM T55959 CO2YH7 137649677 IC50 = 13700 nM T55959 C6YE5R 137649990 IC50 = 16600 nM T55959 C9BJ5L 137650031 IC50 = 63500 nM T55959 CXP2R3 137650379 Ki = 28 nM T55959 C37GZJ 137651008 EC50 > 1000 nM T55959 CJ37YH 137651689 IC50 = 3100 nM T55959 C6GL0F 137652257 IC50 = 292.3 nM T55959 CP9Z8M 137653202 IC50 = 109000 nM T55959 CR9F3Q 137653203 EC50 = 127 nM T55959 C02HUF 137653618 IC50 > 10000 nM T55959 CR25WM 137653998 EC50 = 34 nM T55959 C1JGO6 137654323 IC50 = 2289 nM T55959 CT35OC 137654501 IC50 > 10000 nM T55959 C96BJN 137654642 IC50 = 1390 nM T55959 C46UFA 137654647 IC50 > 10000 nM T55959 CF7M8V 137655321 IC50 = 692.1 nM T55959 CZ6DW1 137655750 IC50 = 283600 nM T55959 CU3DK5 137655842 IC50 = 310 nM T55959 CZ84KG 137656433 IC50 = 317 nM T55959 CQ1SI8 137656684 IC50 = 1704 nM T55959 CZ1XS0 137656786 IC50 = 12800 nM T55959 C56MCJ 137656979 EC50 = 294 nM T55959 C3GX2Z 137657462 IC50 = 43700 nM T55959 C8JO0M 137657681 IC50 = 1500 nM T55959 CSA8G2 137658186 IC50 = 82600 nM T55959 C3XAO8 137658670 IC50 = 4100 nM T55959 CG92PT 137660066 IC50 = 590 nM T55959 CWX6N4 137660247 IC50 = 5040 nM T55959 CEV40N 137661034 IC50 = 940 nM T55959 CLF7V1 137661266 IC50 = 4098 nM T55959 C28EJN 137661323 EC50 = 400 nM T55959 CCSU34 137661732 IC50 = 5180 nM T55959 CS47KN 137662116 IC50 = 1115 nM T55959 COT18S 145011254 Ki = 2440 nM T55959 C9A1VD 145967813 IC50 = 8 nM T55959 CM8TF3 145968603 Ki = 39.81 nM T55959 C4BS6T 145969809 IC50 = 150 nM T55959 CUQ7E0 145970103 Ki = 12.59 nM T55959 CBT6L8 145970391 IC50 = 10 nM T55959 CF67IA 145970695 Ki = 39.81 nM T55959 CB7O9W 145971077 Ki = 158.49 nM T55959 C87MSW 145980271 Ki = 10000 nM T55959 CU53SY 145984002 IC50 > 10000 nM T55959 CU6QS4 145984074 IC50 > 10000 nM T55959 CJ9UZ0 145984374 IC50 = 90 nM T55959 C6I3NT 145984803 IC50 > 10000 nM T55959 C9W6PO 145984940 IC50 > 10000 nM T55959 CT6KH5 145985061 IC50 > 10000 nM T55959 CG2C8H 145985476 IC50 > 10000 nM T55959 C1H2UT 145985812 IC50 > 10000 nM T55959 C5XCV8 145986058 IC50 > 10000 nM T55959 CNJH37 145986752 Ki = 622 nM T55959 CUGO10 145988693 Ki = 1191 nM T55959 CC2G1V 146025727 Ki = 4500 nM T55959 C6P3SR 153287553 Ki > 10000 nM T55959 CV9G7Z 153287572 Ki > 10000 nM T55959 CO85KL 153287574 Ki = 3162.28 nM T55959 C5LXC4 153605593 Ki = 1780 nM T55959 CDN5I4 155510548 IC50 = 4200 nM T55959 CYO17F 155510932 IC50 = 4200 nM T55959 C1TUK0 155512091 IC50 = 7320 nM T55959 CI46AM 155512328 IC50 = 3020 nM T55959 C1Z7ED 155513346 IC50 > 10000 nM T55959 CH4Z9J 155513656 IC50 = 4700 nM T55959 CJPD39 155513983 IC50 = 37800 nM T55959 CJ87WT 155514907 IC50 > 10000 nM T55959 CCF56N 155515030 IC50 = 8300 nM T55959 CCJV20 155515202 IC50 = 6760 nM T55959 CF9PN2 155515352 IC50 = 22400 nM T55959 C5EQD6 155515957 IC50 = 910 nM T55959 C5S7UV 155516776 IC50 = 14000 nM T55959 CB71XT 155517422 IC50 = 6800 nM T55959 CL0T5F 155517981 IC50 = 3800 nM T55959 CPR51V 155519210 IC50 = 63710 nM T55959 CUSA24 155519891 Ki > 10000 nM T55959 CV5H7B 155521007 IC50 = 3590 nM T55959 CRM7H5 155521227 IC50 > 10000 nM T55959 CZLF49 155521764 IC50 > 10000 nM T55959 C20MZN 155522137 IC50 = 28430 nM T55959 CGZ5M1 155522684 IC50 = 6000 nM T55959 CN6LX0 155522764 IC50 = 9580 nM T55959 CO6R3B 155523765 IC50 = 61420 nM T55959 C54HQW 155524272 IC50 = 71590 nM T55959 CWD38V 155524413 IC50 > 10000 nM T55959 CVF9H3 155524550 IC50 = 1430 nM T55959 C8G6HD 155524923 IC50 = 2250 nM T55959 CVF9E8 155525067 IC50 = 19600 nM T55959 CX9PC3 155525160 IC50 = 4100 nM T55959 C3IR8Q 155527001 IC50 = 59740 nM T55959 CHA8R7 155527331 IC50 = 3600 nM T55959 C83RSC 155527543 IC50 = 48090 nM T55959 CFMJ93 155528557 IC50 = 36300 nM T55959 C09MIJ 155528769 IC50 = 22500 nM T55959 C1UTA3 155528931 IC50 = 14640 nM T55959 CJHX15 155529238 IC50 = 2900 nM T55959 CVNK03 155529810 IC50 = 7400 nM T55959 CC6X5O 155530123 IC50 = 1330 nM T55959 C1H5JG 155530980 IC50 = 37700 nM T55959 CVLH72 155531187 IC50 = 650 nM T55959 CMX90R 155531435 IC50 = 24300 nM T55959 CN4P5M 155532365 IC50 = 29390 nM T55959 C2MB4H 155533557 IC50 = 3040 nM T55959 CC26GM 155534211 IC50 = 2300 nM T55959 CQV7D8 155534330 IC50 = 6210 nM T55959 CLTU63 155534741 IC50 = 13500 nM T55959 C0WX1T 155535629 IC50 > 10000 nM T55959 CB79ZW 155536080 Ki = 5011.87 nM T55959 CA25OD 155536376 IC50 = 5300 nM T55959 CRHA67 155536435 IC50 = 1090 nM T55959 CIUS98 155536619 Ki = 6610 nM T55959 C9S2IA 155539605 Ki = 2562 nM T55959 CW37XJ 155543088 IC50 = 2000 nM T55959 C4STU5 155543525 Ki = 497 nM T55959 CA04LZ 155544610 IC50 = 133600 nM T55959 CB1F0Y 155545607 IC50 = 1420 nM T55959 CE5YV0 155545747 IC50 > 10000 nM T55959 CI41YF 155546363 IC50 = 7400 nM T55959 CYOQ12 155546516 IC50 = 5580 nM T55959 C1URC8 155547273 Ki > 10000 nM T55959 CIK5C0 155547331 IC50 = 3850 nM T55959 CFW6O5 155547621 IC50 = 1640 nM T55959 CLH68U 155549829 IC50 > 10000 nM T55959 CAS6B5 155550042 Ki > 10000 nM T55959 CW0EG3 155550602 IC50 = 6970 nM T55959 C0UYA7 155551050 IC50 = 33270 nM T55959 CIJD03 155551639 IC50 = 39500 nM T55959 CNG36O 155553448 IC50 = 2250 nM T55959 CPT82C 155554703 IC50 = 27800 nM T55959 CO9GW3 155554773 IC50 = 2990 nM T55959 C1U2KX 155554780 IC50 > 10000 nM T55959 CH6ZD0 155556044 IC50 > 10000 nM T55959 CIU58J 155556193 IC50 = 3300 nM T55959 C6X2HA 155557651 IC50 = 1470 nM T55959 CM5G9F 155558122 IC50 = 3720 nM T55959 C3E1DP 155558516 IC50 = 1600 nM T55959 CM0WK3 155558540 IC50 = 72480 nM T55959 CQNZ35 155559008 IC50 = 65100 nM T55959 C5B2OZ 155559232 Ki > 10000 nM T55959 C0I1YR 155559387 IC50 > 10000 nM T55959 C28MCV 155559835 Ki > 10000 nM T55959 COK0Q8 155559857 IC50 = 104700 nM T55959 C4O8LX 155560376 IC50 = 4170 nM T55959 CU6YD0 155560597 IC50 = 12200 nM T55959 CZG37L 155565447 IC50 = 65590 nM T55959 C1FJ8G 155565910 IC50 = 5040 nM T55959 C6PR3A 155566487 IC50 = 33000 nM T55959 CN5P9D 155569039 IC50 = 1850 nM T55959 CVUR38 155569643 IC50 = 2480 nM T55959 C3N9VU 10251906 Ki > 500 nM T55959 CP9TR0 10324985 Ki = 407.4 nM T55959 CL6EN1 44276149 IC50 = 9.2 nM T55959 CUKM52 44586281 Ki = 1030 nM T55959 CNG2T7 44586282 Ki = 3490 nM T55959 CP9ED8 44586283 Ki = 3650 nM T55959 COY7T4 44586284 Ki = 1155 nM T55959 CH42YT 45268440 Ki = 12 nM T55959 CVQ56L 70686273 Ki = 18.3 nM T55959 CN10CD 70690421 Ki = 3.79 nM T55959 CGMJ45 70690422 Ki = 2.64 nM T55959 C3M5HI 70690423 Ki = 4.63 nM T55959 CEJ9C6 70690424 Ki = 699 nM T55959 CH0N9M 70690425 Ki = 135 nM T55959 CP82NB 70690426 Ki = 26.9 nM T55959 D00DEH 45483512 Ki = 310 nM T55959 D00FMX 46230706 Ki > 6170 nM T55959 D00GDI 45487890 IC50 = 271 nM T55959 D00HCC 12996705 Ki = 4730 nM T55959 D00KRQ 23113096 Ki = 284 nM T55959 D00QCP 46837647 IC50 = 1065 nM T55959 D00WMS 3047299 IC50 = 2310 nM T55959 D01ABR 44414723 Ki = 1950 nM T55959 D01AOI 44592200 IC50 = 6000 nM T55959 D01EIS 12263801 IC50 > 4000 nM T55959 D01FFX 24691160 IC50 > 7000 nM T55959 D01JYY 11323940 IC50 = 9500 nM T55959 D01MBF 45483536 Ki = 6 nM T55959 D01RWY 44542656 Ki = 709 nM T55959 D01SHR 44593693 IC50 > 10000 nM T55959 D01WWC 16573 Ki > 950 nM T55959 D01YED 45141808 IC50 = 452 nM T55959 D01YNZ 45483529 Ki = 1000 nM T55959 D02DCM 44230874 Ki = 79 nM T55959 D02EKR 3031077 IC50 = 2000 nM T55959 D02ENH 9797657 Ki = 3661 nM T55959 D02ICX 14373 Ki = 8 nM T55959 D02LQG 170832 IC50 = 23 nM T55959 D02NUR 44543266 IC50 = 5600 nM T55959 D02TMK 1614 IC50 = 890 nM T55959 D02YOO 4500 Ki = 30 nM T55959 D02YSN 11651575 IC50 = 4301 nM T55959 D02ZIQ 43227131 IC50 = 852 nM T55959 D03BQV 3033806 IC50 = 3200 nM T55959 D03DQQ 45375938 Ki = 139 nM T55959 D03EMO 16102754 Ki = 23 nM T55959 D03HQF 11644566 IC50 = 167 nM T55959 D03JOX 11311147 Ki = 59.7 nM T55959 D03YQY 46837650 IC50 = 2600 nM T55959 D04KZX 44542809 IC50 = 118 nM T55959 D04NDO 45483400 Ki = 1810 nM T55959 D04NKQ 22599992 Ki = 13 nM T55959 D04ZPF 45483409 Ki = 1080 nM T55959 D05LJC 45483405 Ki = 7370 nM T55959 D05LKO 44414722 Ki = 2940 nM T55959 D05PLF 3031066 IC50 = 1090 nM T55959 D05UMA 10334821 Ki = 550 nM T55959 D05ZUX 44207909 Ki >= 1000 nM T55959 D06CMJ 3127 IC50 = 424 nM T55959 D06EMC 11392888 Ki = 544 nM T55959 D06KNV 3703 Ki = 0.7943 nM T55959 D06LCK 45141805 IC50 = 156 nM T55959 D06QGD 11357862 Ki = 266 nM T55959 D06QIQ 44592241 IC50 = 8800 nM T55959 D06UDU 45483520 Ki = 1680 nM T55959 D06WIV 44578367 Ki = 2470 nM T55959 D07CQD 123692 Ki = 2.2 nM T55959 D07DWS 45483446 Ki > 10000 nM T55959 D07IOX 44543268 IC50 = 135 nM T55959 D07LFR 44231007 Ki = 16 nM T55959 D07OOI 3456 Ki = 3.7 nM T55959 D07PAT 16102753 Ki = 7.8 nM T55959 D07SAA 44543271 IC50 = 265 nM T55959 D07ZOP 11470616 Ki = 51 nM T55959 D08AWN 3058751 Ki = 4544 nM T55959 D08EKQ 46890532 Ki = 2490 nM T55959 D08JCK 16102777 IC50 = 190 nM T55959 D08JLB 45483406 Ki = 1030 nM T55959 D08LAY 13904719 IC50 > 4000 nM T55959 D08MEN 14014889 IC50 > 10000 nM T55959 D08NZE 126280 Ki = 23 nM T55959 D08RCH 44566054 IC50 > 10000 nM T55959 D08SCH 151900 IC50 = 3073 nM T55959 D08SLZ 16102764 Ki = 0.97 nM T55959 D09BYB 45487941 IC50 = 1950 nM T55959 D09FIC 46890395 Ki = 3160 nM T55959 D09IIH 45483459 Ki = 239 nM T55959 D09QZM 11637187 IC50 = 28 nM T55959 D09RPR 16737207 Ki > 10000 nM T55959 D09VTJ 441298 IC50 = 2000 nM T55959 D09XWL 45141379 IC50 = 693 nM T55959 D0A0UC 10244015 IC50 = 128 nM T55959 D0A7GW 45487772 IC50 > 40000 nM T55959 D0B4FN 11148955 Ki = 33.7 nM T55959 D0B5AG 44560576 IC50 = 2000 nM T55959 D0BM0M 44454695 IC50 = 4500 nM T55959 D0BW0V 44589528 Ki > 1400 nM T55959 D0C0GL 3031062 IC50 = 511 nM T55959 D0CG2Y 44133490 Ki = 4310 nM T55959 D0D3QE 11550626 IC50 = 1000 nM T55959 D0E3DM 44592118 IC50 = 15000 nM T55959 D0E6PQ 45483451 Ki = 45 nM T55959 D0EO5P 44414709 IC50 > 4000 nM T55959 D0F5AQ 49798218 Ki = 31.62 nM T55959 D0F6GB 44133853 Ki = 5150 nM T55959 D0G0CJ 45141380 IC50 = 845 nM T55959 D0G1XP 44543273 IC50 = 31 nM T55959 D0G5RH 44462219 IC50 = 23 nM T55959 D0G6BJ 24802842 IC50 = 1.995 nM T55959 D0G8UA 46890321 Ki = 2070 nM T55959 D0GG2J 46890492 Ki > 3160 nM T55959 D0GY8R 45141807 IC50 = 414 nM T55959 D0H2TS 45483528 Ki = 461 nM T55959 D0H4AD 44542509 IC50 = 689 nM T55959 D0HF1N 458519 Ki = 1014 nM T55959 D0I2UC 44230733 Ki = 10 nM T55959 D0I4TO 10107888 IC50 > 10000 nM T55959 D0I7BX 16645664 Ki = 3900 nM T55959 D0I9KV 11220599 IC50 = 39.5 nM T55959 D0IB6Y 11658526 IC50 = 668 nM T55959 D0IC4J 45375937 Ki = 166 nM T55959 D0IR0R 16102751 IC50 = 7.4 nM T55959 D0J4CB 24803184 Ki = 12.59 nM T55959 D0J5AR 11672904 IC50 = 565 nM T55959 D0J5EF 215051 IC50 = 1460 nM T55959 D0J8LQ 607810 Ki = 92 nM T55959 D0K3EW 49799108 Ki = 1.259 nM T55959 D0K6ZT 44133851 Ki > 6180 nM T55959 D0KT2M 44133674 Ki = 6410 nM T55959 D0L0AY 11506691 IC50 = 513 nM T55959 D0L4HU 10084369 IC50 = 127 nM T55959 D0L5MW 181743 Ki > 10000 nM T55959 D0L6RY 11322641 Ki = 82 nM T55959 D0L7BK 44414856 IC50 = 400 nM T55959 D0M3TK 45483431 Ki = 4420 nM T55959 D0M6UK 91827366 IC50 = 6100 nM T55959 D0N0TQ 11571886 IC50 = 147 nM T55959 D0N2KU 44517677 Ki = 2290 nM T55959 D0N2RJ 45483432 Ki > 7000 nM T55959 D0N3DD 105056 Ki = 35.48 nM T55959 D0NC3P 117443 IC50 = 12000 nM T55959 D0NM1F 45487774 IC50 > 14000 nM T55959 D0NY4W 11152502 IC50 = 32 nM T55959 D0O2LC 44543272 IC50 > 100 nM T55959 D0O9BL 11210506 IC50 = 52 nM T55959 D0P6SY 14595987 IC50 > 10000 nM T55959 D0P9EO 45141381 IC50 = 842 nM T55959 D0Q6SH 45483408 Ki = 1450 nM T55959 D0Q8IQ 43794735 IC50 = 1534 nM T55959 D0R1AE 44332186 IC50 = 145 nM T55959 D0R2BM 45268750 Ki = 5 nM T55959 D0R3TA 45483407 Ki = 9120 nM T55959 D0R5AD 43227726 IC50 = 1744 nM T55959 D0R8EV 3027752 IC50 = 209 nM T55959 D0R8TH 16102750 Ki = 37 nM T55959 D0RT9B 11506733 IC50 = 313 nM T55959 D0S1XC 25224941 Ki = 60 nM T55959 D0S4JT 45483466 Ki = 701 nM T55959 D0S9AY 44592244 IC50 = 24000 nM T55959 D0S9IO 44454825 IC50 > 10000 nM T55959 D0SN6R 44592197 IC50 = 1000 nM T55959 D0T2RY 9948320 Ki >= 1000 nM T55959 D0T5VG 11514389 IC50 > 10000 nM T55959 D0T8BU 13904714 IC50 = 1400 nM T55959 D0U3SB 45141806 IC50 = 750 nM T55959 D0U7OD 16043230 IC50 > 400 nM T55959 D0V0PR 45483527 Ki = 396 nM T55959 D0V5GB 11637190 Ki = 38.02 nM T55959 D0V8IZ 44543267 IC50 = 69 nM T55959 D0VY9K 45141809 IC50 = 10000 nM T55959 D0W8BJ 44560674 IC50 = 600 nM T55959 D0W8YO 46230654 Ki = 278 nM T55959 D0W9JK 11220185 IC50 = 744000 nM T55959 D0WB6P 46227262 Ki = 3549 nM T55959 D0X3CF 442879 IC50 = 8350 nM T55959 D0X8GC 45487773 IC50 > 40000 nM T55959 D0X8LG 11243002 Ki = 20.1 nM T55959 D0XF5P 44592119 IC50 = 3800 nM T55959 D0XY9E 3029724 IC50 = 56 nM T55959 D0Y1MJ 16102749 IC50 = 22 nM T55959 D0Y3BI 11572135 IC50 = 463 nM T55959 D0Y5CG 45483467 Ki > 2000 nM T55959 D0Y7CS 44543118 IC50 = 1470 nM T55959 D0Y8UC 3929516 Ki = 13.8 nM T55959 D0YZ3E 44435200 Ki = 3300 nM T55959 D0Z4UF 10524711 Ki = 18 nM T55959 D0Z5GR 46230818 Ki > 6320 nM T55959 D0Z6YA 11289879 IC50 > 4000 nM T55959 D0Z9OX 44414719 IC50 = 1300 nM T55959 D0ZC3Q 44230732 Ki = 11 nM T55959 D0ZE4C 45141608 IC50 = 2270 nM T55959 D0ZU5W 22615724 EC50 = 5210 nM T01908 CGN48U 9827867 IC50 > 2500 nM T01908 CW1G9B 10672666 IC50 > 2500 nM T01908 CW7Q2U 10895700 IC50 > 2500 nM T01908 CIQH43 11445130 IC50 = 220 nM T01908 C37MRI 16718808 IC50 = 530 nM T01908 CVO5L6 24748791 IC50 = 720 nM T01908 C30CFX 44436704 IC50 > 2500 nM T01908 CW5V7Y 44559839 Ki = 1600 nM T01908 C7LJ1C 52941945 IC50 = 3400 nM T01908 CM83VP 72163524 IC50 > 2500 nM T01908 CWP85J 87360663 IC50 > 10000 nM T01908 CJ6DA9 127028140 IC50 = 2440 nM T01908 CD9KI3 127028141 IC50 = 3020 nM T01908 CDQ62V 137637214 Ki > 50000 nM T01908 C2K8JV 137639385 Ki = 10000 nM T01908 CNX46H 137654508 Ki = 10000 nM T01908 D05FYR 11700955 Ki = 1410 nM T32578 CY9A0M 66065 IC50 = 208 nM T32578 CWMH72 54768028 IC50 = 18900 nM T32578 C9DGW0 54768030 IC50 = 5800 nM T32578 C9VEX8 137656890 IC50 = 20500 nM T86679 D06IAR 60961 EC50 = 23500 nM T86679 D09AMZ 1676 Ki = 4700 nM T86679 D09QEI 4740 Ki = 5180 nM T86679 D0B3HD 2519 Ki = 10000 nM T86679 D0F8RA 2153 Ki = 2700 nM T86679 D0R4UW 449193 IC50 > 1000 nM T86679 D0XE1C 219024 EC50 = 10000 nM T86679 D00OAU 9869857 EC50 = 51 nM T86679 D00SUK 216466 Ki = 90 nM T86679 D02YQO 10668061 Ki > 10000 nM T86679 D03OQI 11618368 Ki = 700 nM T86679 D06MIQ 9910098 EC50 = 10000 nM T86679 D07TEP 10117987 Ki > 1000 nM T86679 D0F4ZY 5311037 Ki = 1800 nM T86679 D0F5UN 9953065 Ki = 3981 nM T86679 D0G4CF 11270783 Ki = 8.3 nM T86679 D0L5VS 6448585 IC50 = 1500 nM T86679 D0M2TS 71600087 IC50 = 2600 nM T86679 D0U0KR 3035850 Ki > 10000 nM T86679 D0X0IY 64627 Ki = 269 nM T86679 D0Y6ZK 123683 EC50 = 31.62 nM T86679 D0Z3PO 21874557 Ki = 63 nM T86679 D08ECB 11716665 Ki = 17 nM T86679 D0I5VA 11248240 EC50 >= 10000 nM T86679 D0CH7Z 128784 Ki = 18.9 nM T86679 D00YSJ 158795 Ki = 227 nM T86679 D01VPK 6439091 IC50 = 980 nM T86679 D07ESH 176408 Ki = 1110 nM T86679 D0E4WF 439176 Ki = 8200 nM T86679 D0I7BL 65269 Ki = 47300 nM T86679 D0J2UW 3086599 EC50 = 39.81 nM T86679 D0V5DX 9884817 Ki = 31622.78 nM T86679 D0Y6GJ 176407 Ki = 19.3 nM T86679 CF92BM 45482610 EC50 > 10000 nM T86679 C3CJS6 1330 Ki = 250 nM T86679 C8C2FV 1882 Ki = 1390 nM T86679 CT8UK0 22375 Ki = 23500 nM T86679 CW4V5F 69550 Ki = 27600 nM T86679 CKF52M 71593 Ki > 30000 nM T86679 C3S8KF 76011 Ki = 5620 nM T86679 C6A3PT 95028 Ki = 19400 nM T86679 C3SPQ5 95121 Ki > 30000 nM T86679 C2CG8M 98567 EC50 = 45000 nM T86679 C4VE6D 99562 Ki = 4130 nM T86679 CSV20Q 99619 Ki = 23500 nM T86679 CTJ64S 101422 Ki = 9460 nM T86679 C6OGM1 131432 EC50 = 3490 nM T86679 CU7A5O 149362 EC50 = 145 nM T86679 CK4VZ8 152034 Ki = 6240 nM T86679 CL08HI 185566 Ki > 30000 nM T86679 CA6E5H 215492 EC50 = 948 nM T86679 CD0MT5 215610 EC50 = 54000 nM T86679 CKI18O 217940 Ki = 14500 nM T86679 CFGE25 265603 Ki = 6940 nM T86679 CMH1F9 308531 Ki = 7790 nM T86679 CSZ1R6 317946 Ki = 1660 nM T86679 CU15FG 350741 Ki = 20800 nM T86679 CLZE79 386674 IC50 = 54.3 nM T86679 CW4FT7 395949 Ki = 316.23 nM T86679 C58QWF 456309 Ki = 7072 nM T86679 CYE04Q 541615 Ki = 16.3 nM T86679 C8O7DR 541759 Ki = 3.71 nM T86679 C9GZ0J 541903 Ki = 141 nM T86679 CE9CN4 571407 EC50 > 1000 nM T86679 CCTU50 613506 Ki = 585 nM T86679 CSV78R 626711 IC50 > 30000 nM T86679 CV2D4A 640847 Ki = 19 nM T86679 C1PHA8 655439 Ki = 39.6 nM T86679 C7HKX6 658709 EC50 > 1000 nM T86679 COW21P 750351 Ki = 288 nM T86679 C8Y4NV 851050 Ki > 10000 nM T86679 CC94MT 851051 Ki > 10000 nM T86679 CCM2J1 851052 Ki > 10000 nM T86679 CNJC61 853426 Ki = 220 nM T86679 CHJV30 906099 IC50 > 1000 nM T86679 C5QFM2 933735 Ki > 10000 nM T86679 CK5FB9 935972 Ki = 60.7 nM T86679 CWME72 982689 Ki > 1000 nM T86679 C8ZM4G 1241166 Ki = 337 nM T86679 CM80QJ 1509337 Ki = 190 nM T86679 CW2H9O 1898787 EC50 > 1000 nM T86679 CLU5E8 1899510 EC50 > 1000 nM T86679 CXB0U5 2732424 Ki = 6247 nM T86679 CJ1LX4 2748280 Ki = 608.4 nM T86679 CK8T0W 2748282 Ki = 10.2 nM T86679 C8N2TF 2748294 Ki = 40.8 nM T86679 CW3Z7Q 2814825 Ki > 1000 nM T86679 CD84EF 2817023 Ki = 380 nM T86679 CYEW83 2867529 Ki = 2159 nM T86679 C51GNW 2874872 Ki = 23.6 nM T86679 CG35DP 2882039 Ki = 1811 nM T86679 C6MB7N 2895908 Ki = 1103 nM T86679 CHWU72 2910343 Ki > 30000 nM T86679 CA3P4V 2980395 Ki = 484.6 nM T86679 CS6Q9H 2989397 IC50 > 30000 nM T86679 CRO73B 2989630 Ki = 10000 nM T86679 CWMB15 3042985 EC50 = 45000 nM T86679 C5TCF2 3044933 EC50 = 29000 nM T86679 CBM9N7 3071852 EC50 = 3420 nM T86679 CC48UQ 3162481 Ki > 1000 nM T86679 CPNR09 3162488 Ki = 10000 nM T86679 C2GE9F 3162506 Ki > 1000 nM T86679 C4ZI9K 3162667 IC50 > 1000 nM T86679 CH5L8S 3359650 Ki > 1000 nM T86679 CANG93 3909843 Ki = 12.03 nM T86679 CNM2X6 4675559 Ki = 6544 nM T86679 C70ILQ 5033052 Ki > 1000 nM T86679 C1WDY8 5053422 Ki = 11400 nM T86679 CB6W3I 5130381 Ki = 1572 nM T86679 CC0P2D 6032251 Ki = 1000 nM T86679 CTK1P2 6439089 Ki = 60 nM T86679 C5L8EP 7214067 Ki > 1000 nM T86679 C2TX5N 7315332 Ki > 1000 nM T86679 C32LEZ 9497523 Ki = 75 nM T86679 CTIV02 9794423 Ki = 9480 nM T86679 CKNT38 9801343 Ki = 261 nM T86679 C2EJD7 9803992 Ki > 10000 nM T86679 C92LUT 9805713 Ki = 12100 nM T86679 C6M4HR 9806649 Ki = 3.34 nM T86679 CTC76E 9807634 Ki = 33.7 nM T86679 C98ERU 9814428 Ki = 153 nM T86679 C0JI5S 9819926 Ki > 100000 nM T86679 CVLM89 9821879 Ki = 11 nM T86679 C0TS3U 9822488 Ki = 1 nM T86679 C2O9IQ 9822747 Ki = 205 nM T86679 CAQS87 9824812 Ki = 1715 nM T86679 CK0FX6 9825550 Ki = 1.48 nM T86679 CO51GB 9827315 Ki = 2.291 nM T86679 CUG62V 9827467 Ki = 7.75 nM T86679 C9BZC8 9836304 Ki = 1778 nM T86679 CS6IN9 9839378 Ki = 9 nM T86679 CFXZ58 9839545 IC50 = 2214 nM T86679 C4TOH3 9841364 IC50 = 63 nM T86679 C25KVI 9842054 IC50 = 23 nM T86679 C7HAP8 9843843 Ki > 10000 nM T86679 CUYI26 9844693 Ki = 100 nM T86679 C6XHU0 9846447 Ki = 1.78 nM T86679 CRLO45 9850648 EC50 >= 10000 nM T86679 C2F8KA 9850900 Ki = 9.88 nM T86679 CUB8T7 9857266 Ki = 258 nM T86679 CUZL86 9857422 Ki = 164 nM T86679 CP50JH 9857698 Ki = 254 nM T86679 CUO04X 9857735 Ki = 123 nM T86679 CYXI30 9858577 Ki = 423 nM T86679 C6IK1X 9858578 Ki = 271 nM T86679 CUGV50 9860013 Ki = 865 nM T86679 CV19SJ 9868763 Ki = 58 nM T86679 CRJ04W 9868991 Ki = 81 nM T86679 C7ARK4 9870396 Ki = 22 nM T86679 CQR53Y 9870718 Ki = 2.74 nM T86679 CG47TN 9870719 Ki = 4.92 nM T86679 CR2S4Q 9871761 Ki = 15.2 nM T86679 CQ0T4V 9880392 Ki = 248 nM T86679 CYPJ74 9880921 Ki = 383 nM T86679 CZN50C 9887859 Ki = 200 nM T86679 CLIE16 9890003 Ki = 450 nM T86679 C7C5VN 9890439 Ki = 14 nM T86679 CY71UN 9892149 Ki = 3.65 nM T86679 C8LSD7 9893136 Ki = 41000 nM T86679 C0RCP7 9901171 Ki = 270 nM T86679 CDPV97 9901196 Ki = 10 nM T86679 CW8PY4 9901260 Ki = 109 nM T86679 CJKD76 9901497 Ki = 630 nM T86679 CW8Z9K 9901700 Ki = 643 nM T86679 CTU57Q 9902350 IC50 > 10000 nM T86679 CA52RY 9902562 Ki = 199 nM T86679 CJ3OC1 9902563 Ki = 53 nM T86679 C7YM0O 9904456 Ki = 10.3 nM T86679 CUG70S 9906178 Ki = 139000 nM T86679 CR4SN0 9910158 Ki = 150 nM T86679 CDN1R5 9910926 Ki = 57 nM T86679 CC9FE0 9912816 Ki = 2.04 nM T86679 CO9S7Q 9912946 Ki = 469 nM T86679 CQCI74 9915751 Ki = 43.4 nM T86679 CMGL57 9923269 Ki = 141 nM T86679 C7X1TD 9929470 Ki = 222 nM T86679 C1R8JD 9930130 IC50 = 12 nM T86679 C8TMY5 9932840 EC50 = 1100 nM T86679 CJ5YV8 9935943 Ki = 16.1 nM T86679 CY82JD 9936058 Ki = 26.6 nM T86679 CR05XW 9936467 Ki = 3.93 nM T86679 CW4NR7 9945226 Ki = 160 nM T86679 CL3MY6 9946338 Ki = 879 nM T86679 CBZG96 9949541 Ki = 112 nM T86679 C4MSO1 9950776 Ki = 430 nM T86679 C9F7BL 9953799 Ki = 245 nM T86679 CS23VQ 9954406 Ki = 127 nM T86679 C2KD6M 9954747 EC50 = 1440 nM T86679 C8WR2V 9955052 Ki = 116 nM T86679 C7GH6I 9957239 Ki = 199 nM T86679 CPGT28 9967620 Ki = 646 nM T86679 C2UF7H 9968253 Ki = 907 nM T86679 CDM42Y 9970296 Ki = 42 nM T86679 CMZ6X7 9970667 IC50 = 58 nM T86679 CZE6O5 9975036 EC50 = 10 nM T86679 C5SZL7 9978117 EC50 = 6200 nM T86679 C06EVM 9995603 Ki = 229 nM T86679 CJ83TP 9999033 EC50 > 100000 nM T86679 CMP5T0 10007115 Ki = 20 nM T86679 CPAT84 10020580 EC50 = 100000 nM T86679 CA4X5Z 10026670 Ki > 10000 nM T86679 C9E4GW 10029879 Ki = 21 nM T86679 CLRM29 10046145 Ki = 2900 nM T86679 C3X1QT 10050031 Ki > 10000 nM T86679 CR0OB2 10050439 Ki = 5.4 nM T86679 CQ6ID4 10051061 Ki = 26 nM T86679 C9SM7V 10052252 Ki = 1680 nM T86679 CGE17I 10065148 Ki = 69 nM T86679 C6VLS0 10075248 Ki = 1.3 nM T86679 C4B8TP 10085373 Ki = 394 nM T86679 CFI6P8 10126989 IC50 = 33 nM T86679 C78NYU 10131882 IC50 > 10000 nM T86679 C1AU0B 10150517 Ki = 18 nM T86679 CV87WF 10153029 IC50 = 18 nM T86679 CZ17TE 10153190 Ki > 1000 nM T86679 CBY63V 10155413 Ki = 259 nM T86679 C7OC0T 10156654 IC50 > 10000 nM T86679 C7J5EN 10158974 Ki = 6.026 nM T86679 CRVU75 10164201 Ki = 220 nM T86679 C4FNY6 10175278 Ki = 108 nM T86679 CUC8Y6 10196060 IC50 = 7 nM T86679 C5NOP9 10196114 Ki = 50 nM T86679 C1NW4L 10196517 IC50 = 12 nM T86679 C84MZR 10204847 Ki = 9.333 nM T86679 C9KP1Y 10218183 IC50 = 4 nM T86679 CN9W0F 10225178 Ki = 30 nM T86679 C6A8EB 10237267 IC50 = 15 nM T86679 C84YAW 10237847 IC50 = 12 nM T86679 CZE01H 10238677 IC50 = 17 nM T86679 CP7K3D 10246959 Ki = 5 nM T86679 C5RKX3 10247091 EC50 > 100000 nM T86679 C2HVY5 10248379 EC50 > 100000 nM T86679 CH7VN4 10249674 Ki > 10000 nM T86679 C0TXB5 10250190 EC50 > 100000 nM T86679 CGMN21 10254700 Ki = 3570 nM T86679 CT41UJ 10256007 Ki = 2715 nM T86679 CF1UN5 10267860 Ki = 885 nM T86679 CB5DN6 10288169 IC50 = 14 nM T86679 CH6ZC0 10288197 IC50 = 18 nM T86679 C40WZO 10296638 Ki = 22 nM T86679 CI2E8K 10308937 Ki = 13 nM T86679 CU17KP 10310578 IC50 = 17 nM T86679 C8BO9X 10310768 Ki = 23 nM T86679 CC21BD 10311222 IC50 = 16 nM T86679 CBSE14 10311510 Ki = 127 nM T86679 C0H5MU 10316176 Ki > 10000 nM T86679 CXY40F 10318983 Ki > 10000 nM T86679 CF5N9O 10339165 IC50 = 270 nM T86679 C7IPE9 10346511 Ki = 5010 nM T86679 CHZ32J 10377463 Ki = 13.18 nM T86679 CS1V8I 10379032 Ki = 37 nM T86679 C5HPZ3 10387088 Ki = 48 nM T86679 C5F4WP 10403711 EC50 = 5300 nM T86679 C4UX5I 10404217 Ki = 24 nM T86679 C4LMK8 10421804 Ki = 520 nM T86679 CWUB34 10431614 Ki = 128 nM T86679 CO4H0C 10436433 EC50 = 680 nM T86679 CXOL94 10438449 Ki > 10000 nM T86679 CSD86M 10449535 EC50 = 33000 nM T86679 C8XFL5 10449783 IC50 = 15 nM T86679 C9FQ6C 10452788 Ki = 1.2 nM T86679 CK9FA7 10453097 Ki = 226 nM T86679 CM4C2X 10455080 EC50 = 730 nM T86679 CGM46Y 10455852 EC50 = 960 nM T86679 CJ0U1M 10474279 IC50 = 2400 nM T86679 CHC23X 10505816 Ki = 802 nM T86679 CFOS68 10539663 IC50 = 20.4 nM T86679 CA2BP3 10544916 IC50 = 14 nM T86679 CCD47O 10550242 IC50 = 5830 nM T86679 CNF82D 10563436 Ki = 34 nM T86679 C2S8TH 10577289 IC50 = 1770 nM T86679 CL23DC 10580789 Ki > 10000 nM T86679 CEW4T3 10587109 Ki = 90 nM T86679 C1P5DO 10597086 IC50 = 1900 nM T86679 C02GZY 10601859 Ki = 226 nM T86679 CS2VT6 10605011 Ki = 1861 nM T86679 C2N5UX 10616023 IC50 = 150 nM T86679 CLH03M 10616222 IC50 = 2650 nM T86679 CJ06HI 10618828 IC50 = 77 nM T86679 C8N0QS 10621771 IC50 = 5600 nM T86679 CPLR23 10621961 IC50 = 7400 nM T86679 C8JB3I 10623248 Ki = 303 nM T86679 CC3X4J 10624626 Ki = 1760 nM T86679 CY6QP1 10626463 Ki > 10000 nM T86679 C7QWO6 10637742 Ki = 53 nM T86679 C78YHS 10641040 IC50 = 10 nM T86679 C90VMP 10645103 IC50 = 645 nM T86679 CF0ZO5 10645984 IC50 = 2080 nM T86679 C8O2UT 10647227 Ki = 70 nM T86679 C2NPD5 10648228 Ki = 5.42 nM T86679 CBI7X5 10659581 Ki = 65 nM T86679 C8NCG3 10661707 Ki = 400 nM T86679 C0U2LA 10665761 IC50 = 140 nM T86679 C17GBZ 10669778 IC50 = 250 nM T86679 CGU6W0 10687707 IC50 = 3200 nM T86679 C5RMA3 10688700 EC50 = 32000 nM T86679 CWJ60V 10691124 IC50 = 49 nM T86679 CQV6Y1 10691504 IC50 = 2410 nM T86679 C9B1PF 10696675 Ki = 90 nM T86679 C1XMZ9 10714900 IC50 = 500 nM T86679 CBK4G2 10717193 IC50 = 3660 nM T86679 C07JSG 10720065 Ki = 2.47 nM T86679 C7NXS3 10737168 Ki = 49 nM T86679 CB0L1T 10745111 Ki > 1000 nM T86679 CUG21I 10761800 IC50 = 72 nM T86679 CCZ4U8 10765059 Ki = 2030 nM T86679 CL6VU1 10766773 IC50 = 13300 nM T86679 CK0C8P 10767043 Ki = 2.22 nM T86679 C5B6KP 10769581 Ki = 1113 nM T86679 C3GJ5Z 10779327 Ki = 39 nM T86679 C79MNZ 10791347 Ki = 81 nM T86679 CYG2J5 10792296 Ki = 2.14 nM T86679 C4PK2F 10812045 IC50 = 127 nM T86679 C7BT0O 10824674 IC50 = 15.3 nM T86679 C6UP5K 10834513 Ki = 4294 nM T86679 C2E6PX 10839228 Ki = 16.7 nM T86679 C20WTU 10839296 Ki = 1.52 nM T86679 C89OKC 10840167 Ki = 2.35 nM T86679 C6CSZ4 10852375 Ki = 12 nM T86679 CE04SL 10852506 Ki = 9.1 nM T86679 C3I2WZ 10859484 Ki = 81 nM T86679 CR40LK 10861697 Ki = 691 nM T86679 C3QWZ1 10862463 EC50 > 100000 nM T86679 CZ7WJ9 10863425 Ki = 40 nM T86679 COX52I 10863622 Ki = 6.5 nM T86679 CRU6I1 10863910 Ki = 5.3 nM T86679 C4J8CR 10868826 Ki > 30000 nM T86679 C7RD3K 10872091 Ki > 1000 nM T86679 C4HO6X 10874051 Ki = 24 nM T86679 CB6J8X 10875138 Ki = 1.2 nM T86679 C47HSO 10882425 Ki = 15.1 nM T86679 C1AL7H 10884000 Ki = 31 nM T86679 CN8J0Y 10884265 Ki = 142 nM T86679 CY62BK 10884803 Ki = 305 nM T86679 CIG9Z2 10895416 Ki = 76 nM T86679 C2P1QB 10895565 Ki = 25 nM T86679 CO7S6D 10895702 Ki = 5.5 nM T86679 C2LV6K 10904370 Ki > 1000 nM T86679 CU93CT 10904839 Ki > 10000 nM T86679 C3KOX6 10905184 Ki = 302 nM T86679 CKV30L 10905799 Ki = 50 nM T86679 CH52LS 10906943 Ki = 28 nM T86679 CJ52TM 10916451 Ki > 10000 nM T86679 CS58FH 10917575 Ki = 30 nM T86679 CVFL61 10918042 Ki = 121 nM T86679 CQXA29 10926253 Ki = 12 nM T86679 CCO41S 10926422 Ki = 3.7 nM T86679 C3IA5Y 10927361 Ki = 590 nM T86679 CJB64E 10927693 Ki = 101 nM T86679 CFZ49H 10928011 Ki > 10000 nM T86679 C1B6XL 10928182 Ki = 165 nM T86679 CG2N7W 10928649 Ki = 52 nM T86679 C58CRE 10938276 Ki = 132 nM T86679 CG24MW 10938325 Ki > 10000 nM T86679 C6FQ3L 10938608 Ki = 46 nM T86679 C8BLN4 10939224 Ki = 53 nM T86679 CXWV50 10959335 Ki > 10000 nM T86679 CY2OS9 10961304 Ki = 37 nM T86679 C7YVC5 10962009 Ki > 10000 nM T86679 CA0K1W 10962751 Ki = 2.9 nM T86679 CXH12M 10970127 Ki = 4.4 nM T86679 CD4MO1 10970525 Ki = 13 nM T86679 CLK8M1 10970782 Ki > 1000 nM T86679 CKE84F 10970819 EC50 = 100000 nM T86679 CD16UB 10971099 Ki = 161 nM T86679 C9WLT0 10971427 Ki > 10000 nM T86679 C6OFK0 10971806 Ki = 215 nM T86679 C4ZU8F 10971841 Ki = 161 nM T86679 CBW9J6 10972594 Ki > 10000 nM T86679 C7Z2PT 10980845 Ki = 372 nM T86679 C2TEB7 10981207 Ki = 10.8 nM T86679 C4G0YQ 10982985 Ki = 61 nM T86679 C83XMH 10993869 Ki > 10000 nM T86679 C6BH4T 10993916 Ki = 286 nM T86679 C9NP1R 10994142 Ki > 1000 nM T86679 C3F4TJ 10994183 Ki = 78 nM T86679 CSO19C 10994216 Ki = 35 nM T86679 C31HJV 10994317 Ki = 136 nM T86679 C9IGK2 11003653 Ki = 10000 nM T86679 CMDB43 11004373 Ki = 97 nM T86679 CEP35L 11004986 Ki > 1000 nM T86679 CLR4B8 11005067 Ki > 10000 nM T86679 C0KDE3 11014188 Ki = 165 nM T86679 C47IDH 11014608 EC50 = 100000 nM T86679 C6EQD3 11015003 Ki = 246 nM T86679 C30WTZ 11017082 Ki > 10000 nM T86679 CI3E7D 11019436 Ki > 30000 nM T86679 C8UPZ3 11026001 EC50 = 2600 nM T86679 CF5B8Z 11026358 Ki > 1000 nM T86679 CPD61T 11026434 Ki = 226 nM T86679 C12YXH 11027282 Ki > 10000 nM T86679 CX28EA 11027412 Ki = 25 nM T86679 CW05DS 11028588 Ki > 1000 nM T86679 CHEA89 11037671 Ki > 10000 nM T86679 CR7FM2 11037739 Ki = 87 nM T86679 CM9FK6 11037972 Ki = 296 nM T86679 C5DG1J 11038429 Ki = 14.7 nM T86679 C50MFV 11046203 Ki = 6.8 nM T86679 CS8P0U 11048163 Ki > 10000 nM T86679 CL1RP8 11048438 EC50 = 8900 nM T86679 CW7Q6U 11053743 Ki = 3020 nM T86679 CCS8A6 11058550 Ki = 223 nM T86679 CYZ83I 11059351 Ki = 125 nM T86679 CA91IB 11060260 Ki > 10000 nM T86679 C35IZX 11067937 Ki = 311 nM T86679 CM7TR4 11068963 EC50 = 100000 nM T86679 C9KRQ1 11070905 Ki > 10000 nM T86679 C7HIP2 11071159 Ki = 26 nM T86679 CN5S7E 11078951 Ki > 1000 nM T86679 C1EJI0 11080491 Ki = 31 nM T86679 CKX4G6 11080788 Ki = 150 nM T86679 C4Y7NZ 11081189 Ki = 31 nM T86679 CKEF14 11089092 Ki = 14.5 nM T86679 CR3X1M 11091600 Ki = 45 nM T86679 C64PWO 11091632 Ki = 78 nM T86679 C15EQZ 11091783 Ki = 65 nM T86679 CVDM13 11102838 Ki = 180 nM T86679 CAP6K3 11111247 Ki = 2.7 nM T86679 CMY97P 11112381 EC50 = 100000 nM T86679 C3Z5PU 11112543 Ki = 196 nM T86679 C6RB5D 11112711 EC50 = 9100 nM T86679 C3IFX4 11112849 Ki = 48 nM T86679 CBFQ96 11121771 Ki = 26 nM T86679 CR7X2T 11122708 Ki = 85 nM T86679 CBH3G1 11123022 Ki = 2.5 nM T86679 CLN23H 11123135 Ki > 1000 nM T86679 C06JLD 11123887 Ki > 10000 nM T86679 C4CWA8 11133107 Ki > 1000 nM T86679 CJ86ZM 11133545 Ki = 180 nM T86679 CL19OW 11133804 Ki = 175 nM T86679 CTG5Y7 11133843 Ki = 136 nM T86679 C29UBQ 11143352 Ki = 43.65 nM T86679 CJ47TQ 11143648 Ki = 3.8 nM T86679 CH4TG2 11144119 Ki > 1000 nM T86679 C9N1RL 11144868 Ki = 181 nM T86679 C72QCG 11145314 Ki > 10000 nM T86679 CVF8Z5 11151115 IC50 > 1000 nM T86679 C79YSE 11153187 IC50 > 1000 nM T86679 CM9SW5 11154129 IC50 > 30000 nM T86679 CLQR16 11157262 EC50 = 560 nM T86679 C1FVD5 11162618 Ki = 402 nM T86679 CS0N2C 11164346 EC50 = 9 nM T86679 CPB62L 11174953 EC50 = 19 nM T86679 C12UTW 11175566 IC50 > 1000 nM T86679 CU96ZO 11176782 Ki > 10000 nM T86679 CFL0O8 11177363 IC50 > 30000 nM T86679 CHD65Q 11198201 Ki = 9 nM T86679 CD7QP2 11199731 IC50 > 30000 nM T86679 C41PYH 11209919 IC50 > 1000 nM T86679 C4JK3N 11213889 Ki = 23 nM T86679 C3FP0D 11229946 Ki = 375 nM T86679 C9IHT1 11233411 IC50 > 1000 nM T86679 CB6Y4A 11233413 IC50 > 1000 nM T86679 C7LS3R 11256992 EC50 = 34 nM T86679 CCU71Z 11257069 IC50 > 1000 nM T86679 CL1J5B 11257336 Ki = 3100 nM T86679 C86XNQ 11260448 Ki = 21 nM T86679 CL60TZ 11267343 Ki = 199 nM T86679 C1FT4Y 11282829 Ki = 13 nM T86679 CGR1A8 11289861 Ki = 444 nM T86679 C4PH8A 11306173 Ki = 16 nM T86679 C9KYQ4 11313397 Ki = 8.9 nM T86679 CUS2N9 11313850 Ki = 516 nM T86679 CJX89P 11348709 IC50 > 1000 nM T86679 C3TH4B 11352497 Ki = 624 nM T86679 CRND96 11360082 IC50 > 1000 nM T86679 C8G3FO 11371101 IC50 = 400 nM T86679 CUF53H 11373346 Ki > 1000 nM T86679 CB3J6T 11380878 Ki = 5875 nM T86679 CRU3A7 11381738 Ki = 121 nM T86679 CSD31L 11386134 Ki = 28000 nM T86679 C8KD6J 11386951 EC50 = 1200 nM T86679 CB2C4P 11392671 Ki = 917 nM T86679 CVAJ46 11393155 Ki = 156 nM T86679 CXPM05 11394389 IC50 > 1000 nM T86679 C6IVY0 11408692 Ki = 1913 nM T86679 C61HST 11416002 Ki = 53.4 nM T86679 CCW60O 11420226 Ki = 42 nM T86679 CLD1X7 11420910 Ki = 43 nM T86679 C30ZXP 11426423 Ki = 754 nM T86679 CF4H1A 11428535 IC50 > 1000 nM T86679 C6CV1B 11452333 IC50 > 1000 nM T86679 C5M3SD 11463674 IC50 > 1000 nM T86679 C5JTD0 11464552 IC50 > 1000 nM T86679 C9CFK5 11465677 IC50 > 1000 nM T86679 C9NP2C 11466670 Ki = 48 nM T86679 C9RK6X 11475577 IC50 > 1000 nM T86679 CE7JS1 11483771 Ki = 67 nM T86679 C2SY3I 11492651 Ki > 10000 nM T86679 CI4JC0 11492857 Ki = 3730 nM T86679 CL49IS 11493754 Ki = 2300 nM T86679 CKN80I 11494063 IC50 > 1000 nM T86679 C5FY2G 11494318 Ki = 518 nM T86679 CO32QT 11495161 Ki = 33 nM T86679 C1P7DN 11495410 Ki = 51.29 nM T86679 C29IYG 11495464 Ki > 6600 nM T86679 CH7UC9 11495611 Ki = 20 nM T86679 CNM29H 11495641 Ki = 700 nM T86679 CJ8NX6 11495984 Ki = 22.39 nM T86679 C20ZNT 11496023 Ki = 650 nM T86679 CPIQ63 11497055 Ki = 5.129 nM T86679 C5LN1D 11497238 IC50 = 244 nM T86679 C60KRJ 11498113 Ki = 7.762 nM T86679 C6KL3S 11501678 IC50 > 1000 nM T86679 CD0T6O 11503200 Ki = 58 nM T86679 CQF31J 11503616 Ki = 3.162 nM T86679 CDAC08 11503942 Ki = 20.42 nM T86679 C08TYB 11503979 Ki = 123.03 nM T86679 CL60QU 11505071 Ki = 100 nM T86679 COG79X 11508049 Ki = 9020 nM T86679 C5A8ZL 11508721 Ki = 45.71 nM T86679 C0AWD8 11508923 Ki = 6 nM T86679 C4DUQ1 11509299 Ki = 1513.56 nM T86679 CH3RU8 11510603 Ki > 6600 nM T86679 CSLD98 11510702 Ki = 5.623 nM T86679 CO4B6S 11510891 Ki = 213.8 nM T86679 CLM6Q8 11511593 Ki = 3.162 nM T86679 CI98OZ 11511703 IC50 > 1000 nM T86679 C8GL1J 11511804 Ki > 1000 nM T86679 CYN5U6 11511897 Ki = 250 nM T86679 CH03ZF 11516748 IC50 > 1000 nM T86679 CD29AZ 11517013 Ki > 1000 nM T86679 C56UZA 11517635 Ki = 54.95 nM T86679 CJNF65 11517907 Ki = 19.95 nM T86679 C65MAZ 11519021 Ki = 11.75 nM T86679 CMNY64 11519361 Ki = 83.18 nM T86679 C60VRX 11519405 Ki = 56.23 nM T86679 CT60SW 11522152 Ki > 10000 nM T86679 CS1M7B 11522670 Ki > 30000 nM T86679 CKIR86 11524078 Ki = 79.43 nM T86679 C4K0MX 11524240 Ki = 165.96 nM T86679 CQZ37L 11524264 Ki > 1000 nM T86679 CH9DU2 11524593 Ki = 980 nM T86679 C23LEU 11524637 Ki = 34 nM T86679 CC23GO 11524705 IC50 > 1000 nM T86679 CIJA46 11524904 Ki = 16.98 nM T86679 C1CJ2S 11525283 Ki = 3.62 nM T86679 C3KE4L 11525368 Ki = 13.49 nM T86679 CYAW65 11525776 Ki = 12.59 nM T86679 CIH91Y 11525816 Ki = 20.89 nM T86679 CKC6F5 11529450 Ki = 1440 nM T86679 CR34YL 11530568 Ki = 1548.82 nM T86679 C47MXO 11531253 Ki = 122 nM T86679 C9VYT8 11531274 Ki > 5800 nM T86679 CQSG28 11531275 Ki > 4100 nM T86679 CG49ZV 11531449 Ki = 72.44 nM T86679 CEDZ81 11532717 Ki = 29 nM T86679 C6HAF9 11533237 Ki = 300 nM T86679 C92FYA 11533614 EC50 > 10000 nM T86679 C19JCF 11533636 IC50 > 1000 nM T86679 CAZ51S 11533996 Ki = 6.918 nM T86679 C8P2YI 11536894 Ki > 30000 nM T86679 CU38FS 11537425 Ki = 69 nM T86679 CH43JG 11538373 IC50 > 1000 nM T86679 C5KDX9 11539152 Ki > 10000 nM T86679 CSY78B 11541413 Ki = 8.913 nM T86679 C16FKE 11544506 Ki = 16 nM T86679 CT6C5U 11544894 Ki = 27 nM T86679 CW62MV 11545273 IC50 > 1000 nM T86679 C2QHP4 11545341 Ki = 310 nM T86679 CUD5B0 11546358 IC50 > 1000 nM T86679 C1U8RO 11547107 Ki = 20 nM T86679 C36DPX 11547533 Ki = 186.21 nM T86679 C5NOR2 11548192 Ki = 27.54 nM T86679 CB56MC 11548559 Ki = 12.59 nM T86679 CJ6QB9 11548714 Ki = 24.55 nM T86679 CO28UI 11553439 Ki = 371.54 nM T86679 C3IET8 11553509 Ki = 4.786 nM T86679 C7OJ4E 11554182 Ki = 6.918 nM T86679 C6CVK7 11555032 Ki > 1000 nM T86679 C2NVK8 11555329 Ki = 38.9 nM T86679 CF6E1O 11555462 Ki = 4.074 nM T86679 C0JBI1 11555937 Ki = 77.62 nM T86679 C5RHM0 11555968 Ki = 6.026 nM T86679 CDK2G0 11560108 Ki = 2187.76 nM T86679 C0VES1 11560202 IC50 = 260 nM T86679 C7VD3G 11560510 Ki = 36 nM T86679 C8FM4N 11560981 Ki = 390 nM T86679 C5Q7TL 11561073 Ki = 12.3 nM T86679 CH3TK6 11561715 Ki = 13.8 nM T86679 CI9LM6 11561747 Ki = 79.43 nM T86679 CAN1B7 11562203 Ki = 7.943 nM T86679 C41AXZ 11565780 Ki = 774 nM T86679 CIR70L 11565927 Ki = 116 nM T86679 CV9N6K 11567017 Ki = 102 nM T86679 C5JIZ0 11567699 Ki = 70.79 nM T86679 C93ANH 11568001 Ki = 3.02 nM T86679 CEH5V1 11568060 Ki = 31.4 nM T86679 C9WVP1 11568203 Ki = 14 nM T86679 C85MGW 11568359 Ki = 4.48 nM T86679 C9Y1JH 11568517 Ki = 42.66 nM T86679 CQH34L 11569133 Ki = 34.67 nM T86679 CWUR48 11569515 Ki = 200 nM T86679 CJM06D 11569877 Ki = 33.88 nM T86679 CVY43P 11570614 Ki = 19.5 nM T86679 C54QHO 11574428 Ki = 250 nM T86679 C9VP0G 11574573 EC50 > 10000 nM T86679 C7RA2X 11575498 Ki = 18 nM T86679 CAHB70 11576014 Ki = 16.98 nM T86679 CU3MW5 11576491 Ki = 5.129 nM T86679 CTW85Y 11576751 Ki = 63.1 nM T86679 CX8KA3 11577210 Ki = 131.83 nM T86679 C5JOW8 11580374 Ki > 30000 nM T86679 C8Y9LA 11582537 Ki = 1250 nM T86679 CAR2U3 11582578 Ki = 37 nM T86679 C5I4RZ 11582697 Ki = 18 nM T86679 C8Q3FA 11583705 Ki = 3.162 nM T86679 CB8H3T 11584027 Ki = 10.72 nM T86679 C82YDZ 11584408 Ki = 91.2 nM T86679 C6D1MA 11584660 Ki > 12589.25 nM T86679 COVP09 11584826 Ki = 21.88 nM T86679 C0TFK3 11586663 Ki = 140 nM T86679 CM62BJ 11587409 Ki = 8510 nM T86679 CYJ29E 11587927 Ki = 2530 nM T86679 C8S2RC 11588630 Ki = 19 nM T86679 CU0MX8 11589625 Ki = 28 nM T86679 CR6Y8H 11590025 Ki = 66.07 nM T86679 CH2TN6 11590097 Ki = 27.54 nM T86679 C1L2OW 11590411 Ki = 3.548 nM T86679 C5KX2E 11590453 Ki = 51.29 nM T86679 C9KJ2P 11590537 Ki = 4.898 nM T86679 CE2I5N 11591029 Ki = 19.05 nM T86679 CVE43I 11591558 Ki = 18.62 nM T86679 CI2ZO0 11591823 Ki = 22.91 nM T86679 CS1RK4 11595040 Ki > 10000 nM T86679 CMF50J 11595592 Ki = 43.65 nM T86679 CUXN24 11596614 Ki = 40 nM T86679 C31YOR 11596733 IC50 > 1000 nM T86679 CF3MD9 11597118 Ki = 240 nM T86679 C1QJ4W 11602451 Ki = 5310 nM T86679 C32EKF 11602732 Ki > 6000 nM T86679 C0A4FU 11604435 Ki = 7.762 nM T86679 C21IGF 11608581 Ki = 18 nM T86679 CB06AO 11608818 Ki > 10000 nM T86679 C8LA0I 11609235 Ki > 30000 nM T86679 CWMD07 11610638 Ki = 5 nM T86679 CJW6N3 11610747 Ki = 213.8 nM T86679 C9AQ0O 11610869 Ki = 154 nM T86679 CC6GD1 11611016 Ki = 43.65 nM T86679 CUIT18 11611298 Ki = 15.14 nM T86679 C6NID5 11611580 Ki = 44 nM T86679 C0DGN8 11612118 Ki = 9.55 nM T86679 C2G4JX 11612320 Ki = 37 nM T86679 CE3ZL4 11613517 Ki = 52.48 nM T86679 C39ZVR 11618633 Ki = 100 nM T86679 CCP36O 11618962 Ki = 3.89 nM T86679 C0UO1V 11621020 Ki = 5.888 nM T86679 CLV26W 11623708 Ki = 5790 nM T86679 C7AM8B 11623934 Ki = 3430 nM T86679 C35XDW 11625796 IC50 = 250 nM T86679 CQ2LY3 11627221 IC50 > 1000 nM T86679 C32ECV 11627336 Ki = 3.236 nM T86679 C30LUZ 11627494 Ki = 19.95 nM T86679 C2JW5N 11628044 Ki = 24.55 nM T86679 C0JOM4 11630922 Ki > 10000 nM T86679 CJ5OM1 11632785 Ki = 10.96 nM T86679 CJ02TL 11633189 Ki = 37 nM T86679 C2XD3T 11634901 Ki = 60.26 nM T86679 CFTH84 11638790 Ki = 115 nM T86679 C80FAW 11640539 Ki = 3.802 nM T86679 CRB30J 11640595 Ki = 21.38 nM T86679 CX4V0L 11640619 Ki = 53.8 nM T86679 CG4J8D 11641051 Ki = 263.03 nM T86679 C85ZEB 11642035 Ki = 3.467 nM T86679 CSW2L6 11642231 Ki = 350 nM T86679 CSG21Q 11645609 Ki = 123.03 nM T86679 C9X5JF 11647607 Ki = 35 nM T86679 CE5M6Q 11648670 Ki > 6600 nM T86679 C0GX7S 11649117 Ki = 4.786 nM T86679 C3VZF7 11649145 Ki = 5.248 nM T86679 CV5DW1 11649276 Ki > 5800 nM T86679 CND50M 11649544 Ki = 2.188 nM T86679 CIB32Z 11649548 Ki = 199.53 nM T86679 CAX46N 11654460 Ki = 14 nM T86679 CIS7K1 11654461 Ki = 22 nM T86679 CC8X7R 11655061 Ki = 990 nM T86679 CLU6I0 11656075 Ki = 9.772 nM T86679 CV19DM 11656109 Ki = 410 nM T86679 CJ1X7N 11656185 Ki = 37.15 nM T86679 CFP83C 11656570 Ki = 10.96 nM T86679 CQ8SE2 11656950 Ki = 34.67 nM T86679 CWY7T6 11659363 Ki = 13300 nM T86679 C1JU7A 11659696 Ki = 24 nM T86679 C1JBL4 11660427 Ki = 288.4 nM T86679 C1L0JI 11660995 Ki = 15.85 nM T86679 C4ZB9Y 11661440 Ki = 101 nM T86679 C6OQR7 11662264 Ki = 4800 nM T86679 CV39AR 11662965 EC50 > 10000 nM T86679 C2BH0P 11663050 Ki = 44.67 nM T86679 C7D2CU 11663068 Ki = 4.677 nM T86679 CC9YA7 11664137 Ki = 7.762 nM T86679 CI2SK9 11667107 Ki = 34 nM T86679 CGI6Y3 11667703 IC50 > 1000 nM T86679 C2MW9P 11670078 Ki = 14.13 nM T86679 CV2LY7 11674882 Ki = 269.15 nM T86679 CN04ER 11676113 Ki = 158.49 nM T86679 CAJ43T 11676986 Ki = 26.92 nM T86679 CL6A2N 11677252 Ki = 28.18 nM T86679 C24BUE 11677313 Ki = 3.311 nM T86679 CSTZ64 11677724 Ki = 11.22 nM T86679 CNH01O 11677816 Ki = 8.913 nM T86679 C16PMS 11678491 EC50 > 10000 nM T86679 C7SJI1 11678808 Ki = 17.38 nM T86679 C1I6FC 11680901 Ki > 30000 nM T86679 CKU6E7 11681092 Ki = 6030 nM T86679 CFD86C 11681113 Ki = 11500 nM T86679 CF54VW 11681354 Ki = 9080 nM T86679 CE8WD5 11681429 Ki > 30000 nM T86679 CI8AX3 11683024 IC50 > 1000 nM T86679 C94ZVJ 11683855 Ki = 144.54 nM T86679 CAS80N 11684443 Ki = 2.63 nM T86679 CH30ES 11684672 Ki > 1000 nM T86679 C6UIK7 11684701 Ki = 1.549 nM T86679 CEU52V 11684979 IC50 = 280 nM T86679 CI73GV 11685118 Ki = 173.78 nM T86679 CYFJ70 11687483 Ki = 1040 nM T86679 CT3JM9 11690561 Ki = 13 nM T86679 CI10PQ 11690712 Ki = 4.2 nM T86679 CFJ3X6 11690983 Ki = 25.12 nM T86679 CS9FL1 11693081 Ki = 12.3 nM T86679 CJ68MD 11698623 Ki = 640 nM T86679 CH6Q2D 11698898 Ki = 39 nM T86679 CZ8I6J 11699025 Ki = 25.12 nM T86679 C69PJB 11702501 Ki = 2330 nM T86679 CZ9IX2 11703893 IC50 > 1000 nM T86679 CZE9V5 11705261 Ki = 1 nM T86679 CDG61A 11706151 Ki = 83.18 nM T86679 CR6A2V 11709311 Ki > 30000 nM T86679 CX6E5A 11709650 Ki > 30000 nM T86679 C8KDJ9 11710918 Ki = 27.1 nM T86679 C2LMK1 11711190 Ki = 74 nM T86679 CYI8O4 11711438 Ki > 1000 nM T86679 C72KXO 11711753 Ki = 69.18 nM T86679 C80LHJ 11711754 Ki = 147.91 nM T86679 C6UTA1 11713241 Ki = 360 nM T86679 CPE2Q9 11713242 Ki = 27.54 nM T86679 C3RP8Y 11713561 Ki = 16.22 nM T86679 CIYJ64 11713673 Ki = 60.26 nM T86679 CNR71Y 11717537 IC50 > 1000 nM T86679 CD72OJ 11717832 IC50 > 1000 nM T86679 CCQ78R 11720113 Ki = 12.02 nM T86679 CDZ6P4 11720443 Ki = 141.25 nM T86679 CH5DB1 11720501 IC50 > 1000 nM T86679 CZR29N 11720513 Ki = 13.8 nM T86679 C9J4WY 11728711 Ki > 10000 nM T86679 CAMT16 11728808 Ki = 88 nM T86679 CHM43K 11730776 Ki = 6.1 nM T86679 CR80CF 11731871 Ki > 1000 nM T86679 C5GO4E 11732736 Ki = 161 nM T86679 CHW0A6 11733496 Ki = 35 nM T86679 CG7Y4O 11733556 Ki = 150 nM T86679 CF9Q7M 11733601 Ki = 130 nM T86679 C43GFZ 11739282 Ki = 460 nM T86679 C87SLI 11760836 Ki = 10 nM T86679 CSR32T 11761221 Ki = 241 nM T86679 C7MD4U 11761823 Ki > 10000 nM T86679 CGSN15 11762418 Ki > 10000 nM T86679 CI82XE 11762982 Ki = 30 nM T86679 CT84IV 11774108 IC50 > 1000 nM T86679 C92KBG 11776764 EC50 = 14900 nM T86679 CYU16F 11780616 Ki = 15000 nM T86679 CLPT97 11784369 Ki = 143 nM T86679 C65YJD 11784407 Ki = 70 nM T86679 CGX15W 11793210 IC50 = 160 nM T86679 C6LZ9U 11796362 IC50 = 50 nM T86679 CBZJ16 11798195 Ki = 54 nM T86679 CV7T3H 11798368 Ki = 61 nM T86679 C8ZRL4 11801496 Ki = 2.13 nM T86679 C1ZQF6 11811544 Ki = 251 nM T86679 CPMB38 11811761 Ki = 101 nM T86679 C82LEP 11812897 Ki = 34 nM T86679 C6ANG8 11813241 Ki > 10000 nM T86679 C9KMP8 11822168 Ki = 2330 nM T86679 C4W2ID 11824950 Ki > 1000 nM T86679 C31FGJ 11826577 Ki = 235 nM T86679 C15NOJ 11826924 Ki = 22 nM T86679 CAPF41 11850015 Ki = 7560 nM T86679 C6Y3GI 11952504 Ki = 21 nM T86679 C3Y9JS 11952559 Ki = 11 nM T86679 C9AVS8 11952560 Ki = 23 nM T86679 CD41JX 11952564 Ki = 3 nM T86679 CI6SX1 11952665 Ki = 13 nM T86679 C8OKX0 11952670 Ki = 8 nM T86679 CK3T8W 11953248 Ki = 6 nM T86679 CM0SL3 11956193 Ki = 35 nM T86679 C0KXU5 11977965 Ki > 6000 nM T86679 CXT4S5 11977966 Ki > 6000 nM T86679 CWF2B7 11977967 Ki > 6000 nM T86679 CULI10 11978309 Ki > 6000 nM T86679 C6Z3SF 11978310 Ki > 6000 nM T86679 C1EAC3 11978313 Ki > 6000 nM T86679 CUVN07 11978421 Ki > 6000 nM T86679 CE53IF 11995448 Ki = 505 nM T86679 CUM6T1 11995557 Ki = 207 nM T86679 CF56SH 11995649 Ki = 296 nM T86679 CPF9I3 12066874 IC50 = 1.4 nM T86679 CWFL86 12267225 Ki = 182 nM T86679 CM04PC 12267228 Ki = 457 nM T86679 C3TJI0 12351799 Ki = 513 nM T86679 CRU2O5 12391837 Ki = 289 nM T86679 C2OM1D 12654835 Ki = 8510 nM T86679 CC8Q7D 12766586 IC50 > 30000 nM T86679 CWOQ92 13360944 IC50 > 30000 nM T86679 CWB68X 13525048 Ki = 5530 nM T86679 C3KJN4 13525063 Ki = 11100 nM T86679 C97BVY 13830108 EC50 = 2400 nM T86679 CP59CL 14000474 Ki = 79.6 nM T86679 CD8K6T 14157150 EC50 = 16000 nM T86679 CVS4J0 14426726 Ki = 3210 nM T86679 CENP32 14484978 Ki = 9.75 nM T86679 CHO54J 14978313 Ki = 511 nM T86679 CQ7MK8 15388822 Ki > 30000 nM T86679 CSQ0R5 15388827 Ki > 30000 nM T86679 CEN2O9 15388828 Ki > 30000 nM T86679 CRUI31 15524546 Ki = 206.3 nM T86679 CNI9X7 15578102 Ki = 1660 nM T86679 C1HLX3 15578103 Ki = 2239 nM T86679 CG0I8D 15667089 Ki = 73.2 nM T86679 C8OZ5G 15667105 Ki = 187 nM T86679 CE13QR 15729970 IC50 = 13422 nM T86679 CV8DE2 15729973 IC50 > 30000 nM T86679 CFD31U 15729977 IC50 > 30000 nM T86679 C5GRK6 15729982 EC50 = 33700 nM T86679 C2L4NO 16037920 IC50 = 1 nM T86679 C2Q9UM 16070216 Ki = 63 nM T86679 C8Z2WO 16070220 Ki = 29 nM T86679 C80TJF 16070335 Ki = 11 nM T86679 CQRU95 16070337 Ki = 25 nM T86679 C8E6CH 16070448 Ki = 32 nM T86679 CWFS63 16071777 Ki = 2.2 nM T86679 C36JRA 16071780 Ki = 56 nM T86679 CFN62Q 16071781 Ki = 85 nM T86679 CTIQ90 16071896 Ki = 24 nM T86679 CX2GC6 16071897 Ki = 11 nM T86679 C9K2PE 16071901 Ki = 1 nM T86679 CN7F9X 16072019 Ki = 6 nM T86679 CGX62B 16072020 Ki = 3.5 nM T86679 CL4ON2 16072021 Ki = 2.2 nM T86679 CU42YH 16072022 Ki = 3 nM T86679 CXS8C0 16072023 Ki = 10 nM T86679 CSO1T2 16072024 Ki = 12 nM T86679 CMB8Y9 16078995 Ki = 53.4 nM T86679 C1T7DI 16103162 EC50 > 5000 nM T86679 C87PRE 16103163 EC50 > 5000 nM T86679 C34YIZ 16103164 EC50 > 5000 nM T86679 C6U0TL 16103165 EC50 = 273 nM T86679 CT9O5K 16103166 EC50 > 5000 nM T86679 CA2W9G 16103167 EC50 = 210 nM T86679 CG74XQ 16103168 EC50 = 175 nM T86679 CL87PX 16103169 EC50 = 603 nM T86679 C01PWF 16103170 EC50 > 5000 nM T86679 CO3HF4 16103171 EC50 > 5000 nM T86679 CIAE42 16103176 EC50 = 82 nM T86679 C0Z4KU 16103177 EC50 = 369 nM T86679 C3Y8IU 16103178 EC50 = 227 nM T86679 CA1EH0 16103179 EC50 > 5000 nM T86679 CJ8O9B 16103184 EC50 = 450 nM T86679 CY3R6K 16103185 EC50 = 200 nM T86679 C9F7SM 16103186 EC50 = 340 nM T86679 C7HM0K 16103187 EC50 = 359 nM T86679 C0S1VK 16122818 Ki = 260 nM T86679 CTL0F3 16203668 EC50 = 3270 nM T86679 C4OS0D 16203669 EC50 = 989 nM T86679 CKR25N 16365293 EC50 = 46.77 nM T86679 CZT4J2 16433205 IC50 > 30000 nM T86679 CFE82W 16656768 EC50 > 10000 nM T86679 C7WF2V 16720104 Ki = 119 nM T86679 CT7UO9 16720105 Ki = 39 nM T86679 C9JSW0 16720106 Ki = 28 nM T86679 CMBS67 17198003 Ki = 371.2 nM T86679 CBR05N 17198004 Ki = 3.49 nM T86679 CXRL32 17863158 IC50 > 10000 nM T86679 CL9AX4 17863209 IC50 > 10000 nM T86679 CELB65 17863210 IC50 > 10000 nM T86679 CRWX30 18079460 Ki = 56.6 nM T86679 CAE48W 18171064 Ki = 2968 nM T86679 CF87SP 18440405 Ki = 1490 nM T86679 CX6J0D 18440417 Ki = 2030 nM T86679 CRJ31X 18440425 Ki = 2410 nM T86679 CKE94U 18440431 Ki = 9250 nM T86679 CZO7K8 18440528 Ki = 6300 nM T86679 CH29ON 18440555 Ki > 30000 nM T86679 CU5PX4 19074239 Ki = 7580 nM T86679 CA12QJ 19574107 Ki = 19952.62 nM T86679 CM46VR 19818540 Ki = 9890 nM T86679 CBXA48 20592013 Ki = 211 nM T86679 C5KR4S 20847387 Ki > 30000 nM T86679 C75CPM 21128750 EC50 = 37000 nM T86679 CB2V8H 21603068 Ki > 20000 nM T86679 C25WAJ 21874520 Ki = 937 nM T86679 CTK29C 21874538 Ki = 134 nM T86679 C96PRF 21874571 Ki = 23 nM T86679 C07MZN 21874581 Ki = 741 nM T86679 C5QJC8 21874602 Ki = 593 nM T86679 CXG16I 21874603 Ki = 79 nM T86679 CV2C4F 21874613 Ki = 397 nM T86679 CB7S8A 21874626 Ki = 132 nM T86679 CKG68C 21874634 Ki = 1136 nM T86679 CTX5P2 21874639 Ki = 1294 nM T86679 C1CKS9 21874641 Ki = 84 nM T86679 CU80AG 21874647 Ki = 6 nM T86679 C38CXY 21874661 Ki = 43 nM T86679 C4S5PJ 21874662 Ki = 206 nM T86679 C14FGO 21874668 Ki = 192 nM T86679 C3WLM0 21874675 Ki = 59 nM T86679 COLC85 21874676 Ki = 226 nM T86679 C2PZN3 21874681 Ki = 181 nM T86679 CP84GK 21874685 Ki = 122 nM T86679 CSV0W4 21874686 Ki = 46 nM T86679 CW47EF 21874687 Ki = 225 nM T86679 C3EK0T 21874692 Ki = 440 nM T86679 C3KH4A 21874697 Ki = 24 nM T86679 CDV73C 21874721 Ki = 128 nM T86679 C7GWD4 21874722 Ki = 916 nM T86679 C4L8UK 21874755 Ki = 2110 nM T86679 CLY0E3 21874756 Ki = 118 nM T86679 CWQ47T 21874764 Ki = 443 nM T86679 C74HIZ 21874771 Ki = 634 nM T86679 C7NT1D 21874782 Ki = 88 nM T86679 CG9Y7N 21874786 Ki = 282 nM T86679 C7YRN0 21893339 EC50 = 164 nM T86679 CK4HL6 21916357 Ki = 31 nM T86679 CZRX51 21916371 Ki = 199 nM T86679 CS19AF 21916389 Ki = 7 nM T86679 CBY0E6 21916394 Ki = 22 nM T86679 CI1CO9 21916398 Ki = 60 nM T86679 CZ59CO 21916406 Ki = 21 nM T86679 C2XR0J 21916408 Ki = 21 nM T86679 C03FGL 21916419 Ki = 11 nM T86679 C7Q3RY 21958508 Ki > 6000 nM T86679 CB56UX 21958512 Ki = 26 nM T86679 CBA86P 21958522 Ki = 438 nM T86679 C4I2HN 21958524 Ki = 6 nM T86679 CKQ1C3 21958525 Ki = 28 nM T86679 CBQF27 21958526 Ki = 42 nM T86679 CZI7M9 21958533 Ki > 6000 nM T86679 CZ92NC 21958536 Ki = 38 nM T86679 CFX4B6 21958541 Ki = 255 nM T86679 C2CFG0 21958557 Ki = 19 nM T86679 C1NOM6 21958560 Ki > 6000 nM T86679 CVFZ72 21958565 Ki = 645 nM T86679 CZN1L8 21958583 Ki = 13 nM T86679 CW5NK7 21958593 Ki = 11 nM T86679 C36FJO 21958619 Ki = 6 nM T86679 CG2Z3J 21958639 Ki = 3660 nM T86679 CJ7IB6 21958676 Ki = 526 nM T86679 CTSU04 21958681 Ki = 37 nM T86679 CW5DG9 21958701 Ki = 22 nM T86679 CB2U6L 21958702 Ki = 700 nM T86679 CI9Z8B 21958720 Ki = 5830 nM T86679 CS9R0L 21958721 Ki = 5170 nM T86679 C7RE2I 21958724 Ki = 30 nM T86679 CJO62E 21958725 Ki = 34 nM T86679 C3S7EY 21958726 Ki > 6000 nM T86679 C6F8TR 21958745 Ki = 30 nM T86679 CMF03Z 21958758 Ki = 54 nM T86679 C58MPT 21958761 Ki = 24 nM T86679 C5L8YT 21958762 Ki = 49 nM T86679 C4K7OP 21958764 Ki = 31 nM T86679 CCTJ56 21958775 Ki = 5 nM T86679 CDB0O4 21958780 Ki > 6000 nM T86679 CU7EZ3 21958783 Ki = 13 nM T86679 CUNF42 21958814 Ki = 83 nM T86679 C5HFL6 22002319 Ki = 2490 nM T86679 CFH75K 22002352 Ki > 30000 nM T86679 C02SLQ 22002364 Ki = 13300 nM T86679 CPS61Y 22002375 Ki = 2030 nM T86679 C3CV9X 22002449 Ki = 1110 nM T86679 CKME84 22055296 Ki = 23 nM T86679 C43TSO 22055299 Ki = 36 nM T86679 C7CW3I 22266730 Ki = 73 nM T86679 CZF4S2 22266732 Ki = 24 nM T86679 CTO91Z 22266738 Ki = 82 nM T86679 C75PVI 22266740 Ki = 335 nM T86679 CC2N6M 22266741 Ki = 14 nM T86679 CZL43T 22266742 Ki = 12 nM T86679 C0XT6H 22266744 Ki = 141 nM T86679 CV6E4A 22266746 Ki = 2 nM T86679 CU16OK 22266751 Ki = 15 nM T86679 C4R1WE 22266753 Ki = 120 nM T86679 C2QUH0 22266756 Ki = 48 nM T86679 CLF81K 22266759 Ki = 170 nM T86679 CIOB39 22266761 Ki = 15 nM T86679 CC12SJ 22266763 Ki = 111 nM T86679 C4ZJ1F 22266765 Ki = 21 nM T86679 C3WK8Z 22266766 Ki = 13 nM T86679 CAGC71 22266769 Ki = 25 nM T86679 CV53YM 22266771 Ki = 22 nM T86679 CSC37U 22266775 Ki = 14 nM T86679 CCQ0I1 22266776 Ki = 15 nM T86679 CDWI49 22266778 Ki = 11 nM T86679 CC94DE 22266784 Ki = 64 nM T86679 CPDA63 22283414 Ki = 130 nM T86679 CT4D6I 22446266 Ki = 1720 nM T86679 CJ52EV 23371936 IC50 > 30000 nM T86679 CFT0A1 23371944 Ki > 30000 nM T86679 CO98NZ 23656936 IC50 = 1527 nM T86679 C1SWM6 23657265 IC50 > 1000 nM T86679 CG4I1H 23657266 IC50 > 1000 nM T86679 CLN6I7 23678009 Ki = 70 nM T86679 CRY24K 23702720 Ki = 250 nM T86679 CFE2N1 23757284 EC50 = 220 nM T86679 CVO53U 23900137 EC50 = 2400 nM T86679 CD1C5T 24768447 IC50 > 10000 nM T86679 C90QOD 24768449 IC50 > 10000 nM T86679 C06UBG 24768450 IC50 > 10000 nM T86679 C09WQS 24768452 IC50 > 10000 nM T86679 CK02ZF 24812771 Ki = 145 nM T86679 CY58LE 24827289 EC50 = 289 nM T86679 CGH0U3 24827290 EC50 = 965 nM T86679 C5UO3Z 24827415 EC50 = 174 nM T86679 C32BCU 24827417 EC50 = 143 nM T86679 CKC0W3 24827442 Ki = 11 nM T86679 C0WA2D 24827443 Ki = 46 nM T86679 CQW7H1 24827444 Ki = 22 nM T86679 CIR6E9 24827552 Ki = 45 nM T86679 C15VIG 24827553 Ki = 18 nM T86679 C06PBV 24827554 Ki = 20 nM T86679 C34RNS 24827555 Ki = 16 nM T86679 CGUY42 24827556 Ki = 506 nM T86679 CN1P3A 24827594 Ki = 900 nM T86679 CXD8O5 24827998 Ki = 2536 nM T86679 C2W7YS 24828056 Ki = 42 nM T86679 CWPS95 24828457 Ki = 35 nM T86679 C05BYL 24882472 Ki = 2810 nM T86679 C80WUR 24894016 Ki = 1350 nM T86679 C45DXE 24950690 Ki = 620 nM T86679 CS1ZM6 24950846 Ki = 440 nM T86679 CXRN67 25027416 Ki = 2890 nM T86679 C6ERN5 25027417 Ki = 5820 nM T86679 CCZ72B 25027418 Ki = 6390 nM T86679 CW5YA6 25066016 Ki = 910 nM T86679 CK92QL 25070230 Ki = 158.49 nM T86679 C7JE1V 25147618 IC50 > 1000 nM T86679 C5FHU3 25147619 IC50 > 1000 nM T86679 CN2FL7 25188209 Ki = 836 nM T86679 CB6QZ9 25207803 IC50 = 3.5 nM T86679 CJ0S1U 25230098 IC50 = 495 nM T86679 CN3QA7 25230100 IC50 = 571 nM T86679 CJO09C 25230180 IC50 = 3073 nM T86679 C5PT8L 25230181 IC50 = 18 nM T86679 CH61DM 25230881 IC50 = 39 nM T86679 CE4GZ7 25230948 IC50 = 19 nM T86679 C8W0PI 25230949 IC50 = 32 nM T86679 CCJ16P 25231166 IC50 = 13 nM T86679 C6C5EJ 25231167 IC50 = 120 nM T86679 C3N2CW 25231168 IC50 = 189 nM T86679 CV4CT2 25231169 IC50 = 256 nM T86679 CUI20F 25231170 IC50 = 309 nM T86679 CEG8X7 28622387 EC50 > 1000 nM T86679 CWUA82 42625614 Ki > 10000 nM T86679 C6W4XM 42625615 Ki > 10000 nM T86679 CX8DV9 42625691 Ki > 10000 nM T86679 C5I8NE 42625766 Ki > 10000 nM T86679 CIG29P 42625767 Ki > 10000 nM T86679 CTBW80 42636897 Ki = 2740 nM T86679 C1J6SG 44185870 Ki = 0.406 nM T86679 C3OXF9 44185872 Ki = 0.473 nM T86679 CS9Q4K 44185873 Ki = 11.7 nM T86679 CX24EI 44185874 Ki = 1.99 nM T86679 CWH1S5 44185932 Ki = 7.49 nM T86679 CWX1B7 44185933 Ki = 7.51 nM T86679 CF2K1H 44185934 Ki = 5.43 nM T86679 C8PMD7 44185935 Ki = 19.7 nM T86679 C8I9LD 44185936 Ki = 3.03 nM T86679 CQRH91 44186579 Ki = 1.15 nM T86679 C9RG0P 44186580 Ki = 0.215 nM T86679 C48XKD 44186582 Ki = 0.61 nM T86679 CCNH98 44186622 Ki = 0.782 nM T86679 CY2D4F 44186623 Ki = 1.27 nM T86679 CRWD47 44186624 Ki = 0.595 nM T86679 CAY95F 44186625 Ki = 0.695 nM T86679 C42DUI 44186626 Ki = 0.446 nM T86679 CYE0X8 44186667 Ki = 0.303 nM T86679 CM7B3X 44186668 Ki = 0.281 nM T86679 C69VCO 44186669 Ki = 0.775 nM T86679 CSBP65 44186670 Ki = 1.58 nM T86679 CZJ29Y 44186715 Ki = 0.858 nM T86679 C5X9NC 44186716 Ki = 1.19 nM T86679 C6JG3Q 44186717 Ki = 0.944 nM T86679 CE21OP 44186718 Ki = 0.875 nM T86679 C9W0OQ 44186719 Ki = 1.06 nM T86679 CC35JG 44219683 Ki = 2.884 nM T86679 CXIT13 44219684 Ki = 9.12 nM T86679 CQ01KW 44224278 Ki = 6.5 nM T86679 CD49OQ 44236417 Ki = 83 nM T86679 CKNV96 44236419 Ki = 10.7 nM T86679 CNJ14Q 44236420 Ki = 5 nM T86679 CRE3W9 44236421 Ki = 0.9 nM T86679 C8XVK2 44236445 Ki = 1.8 nM T86679 CKV19T 44236503 Ki = 5.9 nM T86679 CW5XG6 44236505 Ki = 6.3 nM T86679 CL2SC0 44236506 Ki = 12 nM T86679 CM5J9N 44236539 Ki = 1.8 nM T86679 CJ40YS 44236566 Ki = 29 nM T86679 C5JMV3 44236567 Ki = 5 nM T86679 C75UQR 44236568 Ki = 8 nM T86679 CO6Y4M 44236571 Ki = 7.4 nM T86679 C49CVJ 44236600 Ki = 1.5 nM T86679 C5AOR8 44236601 Ki = 5.5 nM T86679 C8JB0I 44236602 Ki = 7.3 nM T86679 C6XIR4 44236603 Ki = 190 nM T86679 C30OLC 44236632 Ki = 14 nM T86679 CI6YL0 44236657 Ki = 17.6 nM T86679 C83WVZ 44236659 Ki = 6.7 nM T86679 C19BQS 44236767 Ki > 1000 nM T86679 C2XN9C 44236850 Ki = 12 nM T86679 CE27HN 44276476 Ki = 1.88 nM T86679 C7T0ZY 44281663 Ki = 95 nM T86679 CX3YV9 44281684 Ki = 649 nM T86679 CJ3QM8 44281700 Ki = 110 nM T86679 CN72HK 44281738 Ki = 58 nM T86679 C3XPZ6 44284710 Ki = 6530 nM T86679 CGV41U 44307827 Ki = 36.7 nM T86679 CZB6V2 44307909 Ki = 21600 nM T86679 C6I1EY 44308015 Ki = 8710 nM T86679 CUAO23 44308307 Ki = 15400 nM T86679 CRKG51 44308394 Ki = 14000 nM T86679 CAD3Q7 44308481 Ki = 59.5 nM T86679 C1WOU3 44308520 Ki = 310 nM T86679 CY4DQ7 44390444 Ki = 2780 nM T86679 C3D6LX 44390522 Ki = 1120 nM T86679 CF6WX2 44390523 Ki = 91 nM T86679 C25RFG 44390527 Ki = 1450 nM T86679 CWR5M2 44390528 Ki = 485 nM T86679 CBZ2P1 44390545 Ki = 215 nM T86679 CEB5I3 44390547 Ki > 6666 nM T86679 CE53OI 44390549 Ki = 1830 nM T86679 CG4KO6 44390551 Ki = 4520 nM T86679 CHZ5D1 44390559 Ki = 325 nM T86679 C6HBX7 44390571 Ki = 945 nM T86679 C6XV9J 44390583 Ki = 557 nM T86679 CLQ41H 44390587 Ki = 2080 nM T86679 CA4KL8 44390599 Ki > 2000 nM T86679 C0XIJ4 44390615 Ki = 1010 nM T86679 CD2F9O 44390651 Ki = 207 nM T86679 C8Q9XH 44390669 Ki > 2000 nM T86679 C4QNR0 44401051 Ki = 18800 nM T86679 CA52CR 44404010 Ki = 4.8 nM T86679 CN94AX 44406328 Ki = 63 nM T86679 C3JPG9 44406334 Ki = 195 nM T86679 C3S9CP 44406397 Ki = 163 nM T86679 CAF1Y3 44406398 Ki = 121 nM T86679 CT21RA 44406403 Ki = 131 nM T86679 CA8FV4 44406545 Ki = 19 nM T86679 CG8MQ9 44406555 Ki = 82 nM T86679 CUPC05 44406556 Ki = 106 nM T86679 C5ZW8S 44406562 Ki = 82 nM T86679 CQ98MC 44406567 Ki = 100 nM T86679 CN7V0Y 44406570 Ki = 123 nM T86679 CI19OT 44406582 Ki = 128 nM T86679 CZPM65 44406588 Ki = 136 nM T86679 C6O9TH 44406592 Ki = 74 nM T86679 CJA23V 44406607 Ki = 38 nM T86679 CV5AO7 44406611 Ki = 14 nM T86679 CE3CP9 44406617 Ki = 42 nM T86679 CVQ2B8 44406625 Ki = 134 nM T86679 CD9E7F 44406639 Ki = 55 nM T86679 CK7GF1 44406642 Ki = 18 nM T86679 CPEV01 44406643 Ki = 32 nM T86679 C9ZY1L 44406891 Ki = 7.943 nM T86679 CXL90H 44406904 Ki > 1000 nM T86679 CR8AU6 44406906 Ki = 186.21 nM T86679 CTHP76 44406920 Ki > 1000 nM T86679 C9XF6Y 44406930 Ki = 5888.44 nM T86679 CK9ZB7 44407518 EC50 > 10000 nM T86679 CES29R 44408316 IC50 = 320 nM T86679 C6E4RA 44410402 Ki = 26466 nM T86679 C5IVA3 44410403 Ki = 5533 nM T86679 CI7W8R 44410406 Ki = 8970 nM T86679 CWQX21 44410409 Ki = 3862 nM T86679 C7DER1 44410550 Ki = 7620 nM T86679 CZ94PN 44410554 Ki = 1188 nM T86679 COWL13 44410555 Ki = 21465 nM T86679 CHU6Q0 44410556 Ki = 23800 nM T86679 CXD2R9 44410566 Ki = 1268 nM T86679 C20FJQ 44410585 Ki = 24057 nM T86679 CQ8E2B 44410597 Ki = 2481 nM T86679 CSTP07 44410691 Ki = 8473 nM T86679 CV37TH 44410697 Ki = 7920 nM T86679 C5RU0V 44412318 Ki > 5800 nM T86679 CV9C5B 44413096 IC50 = 75 nM T86679 CNDQ05 44413106 IC50 = 6 nM T86679 C4W7PD 44413112 IC50 = 10 nM T86679 C7PAD9 44413113 IC50 = 15 nM T86679 C4QER5 44413125 IC50 = 7 nM T86679 C5R8YD 44413130 IC50 = 27 nM T86679 C2DN0P 44413136 IC50 = 43 nM T86679 CZ97OD 44413142 IC50 = 90 nM T86679 CB25JN 44413154 IC50 = 6 nM T86679 C1PI5R 44413182 IC50 = 20 nM T86679 CMT4W9 44413192 IC50 = 15 nM T86679 COK1D7 44413193 IC50 = 17 nM T86679 C2ZH7P 44413202 IC50 = 13 nM T86679 COD4F9 44417680 Ki = 611 nM T86679 CSR4Q2 44420921 EC50 = 1780 nM T86679 CO68UH 44420926 EC50 = 54.5 nM T86679 C3C8LS 44423811 EC50 = 7.3 nM T86679 CWCH32 44423812 EC50 = 15.2 nM T86679 CDY6P7 44423813 EC50 = 12.3 nM T86679 CYR14N 44423814 EC50 = 10.5 nM T86679 C2F3DE 44423815 EC50 = 30.2 nM T86679 CF26JD 44423816 EC50 = 107 nM T86679 CE76XB 44423817 EC50 = 32.4 nM T86679 C5J3PM 44423818 EC50 = 45.4 nM T86679 CA2HW6 44423819 EC50 = 53.6 nM T86679 CFM1I4 44423820 EC50 = 35.5 nM T86679 CFTE30 44423821 EC50 = 16.4 nM T86679 CQL6J8 44423822 EC50 = 300 nM T86679 C4QFX3 44423823 EC50 = 32.3 nM T86679 CWQK67 44423824 EC50 = 150 nM T86679 CG5O9I 44423825 EC50 = 240 nM T86679 CK1EQ6 44423826 EC50 = 315 nM T86679 C4ZL9F 44423827 EC50 = 42.6 nM T86679 CH96WQ 44423828 EC50 = 360 nM T86679 CLJ9T4 44423837 EC50 = 175 nM T86679 CT1YQ4 44423838 EC50 = 302 nM T86679 CBW73G 44430154 Ki > 6000 nM T86679 CDU4P8 44430156 Ki > 6000 nM T86679 CA9L1D 44430158 Ki > 6000 nM T86679 C9M0OF 44430160 Ki > 6000 nM T86679 C0HBJ8 44430163 Ki > 6000 nM T86679 CQF30M 44430165 Ki > 6000 nM T86679 C2F3ZV 44430169 Ki > 6000 nM T86679 C4IT7U 44430170 Ki > 6000 nM T86679 C4S5DC 44430171 Ki > 6000 nM T86679 CYS8I1 44430173 Ki > 6000 nM T86679 CLW6M5 44430177 Ki > 6000 nM T86679 CZ2CX5 44430187 Ki > 6000 nM T86679 C42LMQ 44430188 Ki > 6000 nM T86679 C0UDY1 44430192 Ki > 6000 nM T86679 C87TZB 44430198 Ki > 6000 nM T86679 CI97LW 44430203 Ki > 6000 nM T86679 CPW14D 44430206 Ki > 6000 nM T86679 CNX54A 44430209 Ki > 6000 nM T86679 CC20AB 44430231 Ki > 6000 nM T86679 C09MBQ 44430232 Ki > 6000 nM T86679 CDH26R 44430235 Ki > 6000 nM T86679 C8UN2W 44430236 Ki > 6000 nM T86679 C07JTM 44430237 Ki > 6000 nM T86679 CX5RU6 44430239 Ki > 6000 nM T86679 CL6C1D 44430241 Ki > 6000 nM T86679 C21UTJ 44437214 Ki = 7200 nM T86679 C2S1DI 44437219 Ki = 13400 nM T86679 CAO98V 44437220 Ki = 10000 nM T86679 CJSR20 44437233 Ki > 10000 nM T86679 C67ZNA 44437460 Ki > 1000 nM T86679 CYB86Z 44442015 Ki > 10000 nM T86679 C1UIO8 44442016 Ki > 10000 nM T86679 CUP5T0 44442018 Ki > 10000 nM T86679 C4RDK6 44442019 Ki = 8580 nM T86679 CPC63E 44442162 Ki > 10000 nM T86679 C71XQS 44442163 Ki > 10000 nM T86679 C42ZRD 44442166 Ki > 10000 nM T86679 C9Z3CW 44442167 Ki = 1450 nM T86679 CAZR53 44446475 Ki > 6000 nM T86679 C06RLU 44446477 Ki = 3 nM T86679 CFPZ19 44447519 Ki = 8350 nM T86679 CJ7MS5 44447534 Ki = 30800 nM T86679 C3LOJ1 44447535 Ki = 12100 nM T86679 CME34Q 44449532 Ki = 2479 nM T86679 CZUB58 44449635 Ki = 1560 nM T86679 CHP5W0 44450290 EC50 = 920 nM T86679 CCMZ32 44450517 Ki = 27 nM T86679 C6Y0PD 44450826 Ki = 9.55 nM T86679 C6J4IM 44450828 Ki = 7.244 nM T86679 C6VFH5 44450829 Ki = 8.71 nM T86679 C7UPI4 44450849 Ki = 4.677 nM T86679 CSO5T9 44450850 Ki = 7.586 nM T86679 CFW9U0 44450875 Ki = 891.25 nM T86679 CR79ZP 44450903 Ki = 30.9 nM T86679 CR5BE0 44450904 Ki = 20.89 nM T86679 CU4SW3 44450905 Ki = 21.38 nM T86679 CN38SJ 44450929 Ki = 13.49 nM T86679 CTBV26 44450930 Ki = 11.22 nM T86679 CHU69T 44450931 Ki = 12.3 nM T86679 CJ6D7U 44450932 Ki = 6.918 nM T86679 CA01KF 44450933 Ki = 6.607 nM T86679 CGXZ65 44450955 Ki = 9.12 nM T86679 CD5WU9 44450958 Ki = 9.55 nM T86679 CQ6K2P 44450979 Ki = 6.166 nM T86679 C8XGN7 44450981 Ki = 2.884 nM T86679 C76MCE 44450982 Ki = 5.5 nM T86679 C6PK0V 44450983 Ki = 6.166 nM T86679 CVC48J 44450997 Ki = 2.5 nM T86679 CGW63R 44451018 Ki = 69.18 nM T86679 C76WNY 44451019 Ki = 25.7 nM T86679 CCF1X3 44451020 Ki = 25.7 nM T86679 C5J8RO 44451021 Ki = 4.786 nM T86679 CEN6T1 44451048 Ki = 15.14 nM T86679 CSH7C2 44451049 Ki = 14.79 nM T86679 C0N8UL 44451050 Ki = 13.18 nM T86679 C1J9DN 44451053 Ki = 4.169 nM T86679 CFJN06 44451072 Ki = 7.413 nM T86679 C3F9IW 44451073 Ki = 11.75 nM T86679 C1Z9JQ 44451074 Ki = 6.026 nM T86679 CASC19 44451075 Ki = 1.5 nM T86679 CL4H9C 44451099 Ki = 4.898 nM T86679 CN4GU2 44451100 Ki = 5.754 nM T86679 C40RIL 44451105 Ki = 478.63 nM T86679 CV4I0S 44451106 Ki = 173.78 nM T86679 C4N3OQ 44451123 Ki = 4.266 nM T86679 CNEP36 44451126 Ki = 4.169 nM T86679 CN7TA8 44451127 Ki = 2 nM T86679 C6JO2N 44451128 Ki = 70.79 nM T86679 CHZU82 44451129 Ki = 58.88 nM T86679 C0WE7Z 44451165 Ki = 100 nM T86679 CB5WF8 44451166 Ki = 1 nM T86679 CZB19U 44451169 Ki = 57.54 nM T86679 CPGH68 44451171 Ki = 53.7 nM T86679 CPX20Z 44451197 Ki = 169.82 nM T86679 CXYO54 44451199 Ki = 24.55 nM T86679 CKM13P 44451200 Ki = 38.9 nM T86679 CKIL97 44451201 Ki = 51.29 nM T86679 C75LZM 44451224 Ki = 43.65 nM T86679 CU2Y9G 44451227 Ki = 16.98 nM T86679 CPL9E7 44451229 Ki = 10.47 nM T86679 C52UIJ 44451230 Ki = 20.42 nM T86679 CJEA96 44451252 Ki = 13.18 nM T86679 C8CQ3K 44451253 Ki = 9.55 nM T86679 C2Y9WZ 44451254 Ki = 10.96 nM T86679 CMN2L6 44451269 Ki = 8.128 nM T86679 CUE61I 44451271 Ki = 7.079 nM T86679 C7HMX9 44451272 Ki = 6.31 nM T86679 C50QVJ 44451283 Ki = 5.248 nM T86679 CUA67B 44451284 Ki = 6.31 nM T86679 C74QDH 44451285 Ki = 4.169 nM T86679 C3OM0Y 44451303 Ki = 3.631 nM T86679 CAL31F 44451305 Ki = 3.467 nM T86679 CJO78N 44451306 Ki = 3.388 nM T86679 C9U8GO 44451329 Ki = 1.82 nM T86679 C21QUX 44451330 Ki = 2.818 nM T86679 CMQ4H8 44451480 Ki = 51.29 nM T86679 CEL5J8 44451482 Ki = 32.36 nM T86679 C0ZD4U 44451483 Ki = 31.62 nM T86679 C0TLS7 44451489 Ki = 27.54 nM T86679 CEG1Y5 44451491 Ki = 13.49 nM T86679 CE9Q5B 44451492 Ki = 20.42 nM T86679 C1KXG7 44452431 Ki = 2511.89 nM T86679 C6AG2Y 44452434 Ki = 251.19 nM T86679 CJW91V 44452435 Ki = 501.19 nM T86679 C87QHW 44452454 Ki = 144.54 nM T86679 C0PER5 44452455 Ki = 251.19 nM T86679 CTMF29 44452493 Ki = 2398.83 nM T86679 C6DU3Q 44452514 Ki = 426.58 nM T86679 C18BXC 44452535 Ki = 123.03 nM T86679 CWF9E6 44452536 Ki = 67.61 nM T86679 C8SIX2 44452695 Ki = 1737.8 nM T86679 CR58PU 44457922 Ki > 10000 nM T86679 CIDT05 44457923 Ki > 10000 nM T86679 C0GTF5 44457953 Ki > 10000 nM T86679 C2GTV4 44458220 Ki > 10000 nM T86679 C8E9VG 44459944 Ki = 23200 nM T86679 CB7K2Y 44520941 Ki = 1089 nM T86679 CZ6F9S 44520976 Ki = 3185 nM T86679 CQ71XC 44520980 Ki = 2466 nM T86679 CEO4P7 44520981 Ki > 10000 nM T86679 C31SUP 44520982 Ki = 798 nM T86679 CNR53B 44520983 Ki = 1304 nM T86679 C3MZC5 44520985 Ki = 1844 nM T86679 CJ57RW 44537897 IC50 = 5480 nM T86679 C9SK6P 44551168 Ki = 7.413 nM T86679 CW0B5D 44570367 IC50 > 1000 nM T86679 C9BA3H 44570369 IC50 > 1000 nM T86679 C24CRG 44570413 IC50 > 1000 nM T86679 C6EAT9 44570414 IC50 > 1000 nM T86679 CTS6P4 44570415 IC50 > 1000 nM T86679 CP93SE 44570416 IC50 > 1000 nM T86679 C6NJP3 44570454 IC50 > 1000 nM T86679 CC6TW2 44570455 IC50 > 1000 nM T86679 CG9BR2 44570456 IC50 > 1000 nM T86679 C9FV0G 44570457 IC50 > 1000 nM T86679 CC51RV 44570458 IC50 > 1000 nM T86679 CSMN18 44570493 IC50 > 1000 nM T86679 CMD87Q 44572294 Ki > 30000 nM T86679 CSL0G8 44572353 Ki > 30000 nM T86679 C0ETQ1 44572354 Ki > 30000 nM T86679 C7D2GC 44572410 Ki > 30000 nM T86679 C9VS8P 44572470 Ki > 30000 nM T86679 CDZ14G 44572472 Ki > 30000 nM T86679 C8Y0EI 44574117 Ki = 2.8 nM T86679 CZDG39 44574118 Ki = 9.5 nM T86679 CZX7N5 44574165 Ki = 0.7943 nM T86679 C6TIR8 44574166 Ki = 10 nM T86679 CLTE07 44574167 Ki = 81.3 nM T86679 CJ3LA8 44574168 Ki = 3.2 nM T86679 CWDA90 44574191 Ki = 11.5 nM T86679 C0BP3Z 44574192 Ki = 2.1 nM T86679 CX6KL4 44574193 Ki = 16.2 nM T86679 CUH78B 44574194 Ki = 7.1 nM T86679 CMFB42 44574222 Ki = 2 nM T86679 C4VBL3 44574223 Ki = 501 nM T86679 CSA38M 44574224 Ki = 602 nM T86679 CUBQ21 44574225 Ki = 7.8 nM T86679 CY14AD 44574251 Ki = 1.7 nM T86679 C7GY5T 44574252 Ki = 5.9 nM T86679 C4V5GO 44574254 Ki = 24 nM T86679 CN2OG0 44574281 Ki = 42.7 nM T86679 CF5W7A 44574282 Ki = 13.8 nM T86679 CCB34Q 44582614 Ki > 10000 nM T86679 CSM58E 44582652 Ki > 10000 nM T86679 CA5R4M 44582653 Ki > 10000 nM T86679 CR95SV 44582654 Ki > 10000 nM T86679 C8G4TH 44582690 Ki > 10000 nM T86679 CV5F9X 44582691 Ki > 10000 nM T86679 C71SDJ 44582723 Ki > 10000 nM T86679 CLW60K 44582724 Ki > 10000 nM T86679 CH07JS 44582725 Ki > 10000 nM T86679 CZ91EO 44582726 Ki > 10000 nM T86679 C9Y8VU 44583006 Ki = 53.4 nM T86679 CR3LW0 44583035 Ki = 11 nM T86679 CLZ6A1 44587954 Ki = 338 nM T86679 C6B4KH 44587955 Ki = 35 nM T86679 C6IO7C 44587956 Ki = 1 nM T86679 CUG8E4 44587957 Ki = 2.6 nM T86679 C3FQ9A 44588393 Ki = 68 nM T86679 C6IE2F 44588394 Ki = 676 nM T86679 CG1JD0 44588395 Ki = 54 nM T86679 CV6LB9 44588396 Ki = 589 nM T86679 CNG85D 44588436 Ki = 89 nM T86679 C36UPO 44588437 Ki = 155 nM T86679 C71HQU 44588438 Ki = 19 nM T86679 CD97HM 44588439 Ki = 44 nM T86679 CX7YZ2 44588470 Ki = 115 nM T86679 C5QB8V 44588471 Ki = 11 nM T86679 CWN0S7 44588472 Ki = 490 nM T86679 C4JS6Y 44588473 Ki = 479 nM T86679 C4UT7D 44588474 Ki = 24 nM T86679 CN8Q2U 44588514 Ki = 71 nM T86679 CN0M8J 44588515 Ki = 50 nM T86679 CBL10K 44588516 Ki = 6.5 nM T86679 C0UD5O 44588517 Ki = 64 nM T86679 C83AJU 44588518 Ki = 23 nM T86679 CFIA83 44631910 IC50 > 50000 nM T86679 CV1GD3 45073485 IC50 = 23.5 nM T86679 C24KLI 45267987 Ki = 858 nM T86679 CG7M5U 45267990 Ki = 137 nM T86679 C35COL 45267991 Ki = 20.89 nM T86679 CX67BG 45268854 Ki = 1995.26 nM T86679 C7T3HW 45268867 Ki = 11.75 nM T86679 C1IL3E 45268869 Ki = 184 nM T86679 C9WOM0 45268873 Ki = 48.98 nM T86679 CXI20R 45268920 Ki = 125.89 nM T86679 C8AL4S 45268921 Ki = 85.11 nM T86679 C5I0MX 45268927 Ki = 323.59 nM T86679 C8IM6P 45268928 Ki = 147.91 nM T86679 CU2D9I 45269706 Ki = 77.62 nM T86679 C1YSN9 45269707 Ki = 3.02 nM T86679 CW3QL8 45269711 Ki = 15.49 nM T86679 C5QT0W 45269769 Ki = 70.79 nM T86679 CJP69G 45270541 Ki = 924 nM T86679 C5HQ6O 45270544 Ki = 93.33 nM T86679 CTL27N 45271361 Ki = 3.02 nM T86679 CK52VZ 45271363 Ki = 33.88 nM T86679 CNAT29 45272259 Ki = 15.49 nM T86679 CQ6N7W 45272308 Ki = 138.04 nM T86679 C5YT4Z 45273099 Ki = 489.78 nM T86679 CS4L5G 45273118 Ki = 173.78 nM T86679 C6O8XQ 45273122 Ki = 1240 nM T86679 CPG3L9 45481619 IC50 = 1390 nM T86679 C2ZI4P 45481621 IC50 = 780 nM T86679 CCMX92 45481749 IC50 = 10370 nM T86679 CXM9F4 45481750 IC50 = 363 nM T86679 CBOG84 45481751 IC50 > 10000 nM T86679 CLZV08 45481752 IC50 > 10000 nM T86679 C3MPR1 45481753 IC50 = 8960 nM T86679 CB52VK 45481754 IC50 = 491 nM T86679 C5W4NR 45481755 IC50 > 10000 nM T86679 CQOB79 45481756 IC50 = 9370 nM T86679 CB8NA2 45481757 IC50 = 15000 nM T86679 CL68UB 45481758 IC50 = 13700 nM T86679 CY2WO6 45481759 IC50 = 8960 nM T86679 CV43FT 45481760 IC50 = 5840 nM T86679 C50HVN 45481761 IC50 = 11100 nM T86679 C4C0QV 45481762 IC50 > 10000 nM T86679 C16LEJ 45481763 IC50 > 50000 nM T86679 C1TB7C 45481764 IC50 > 10000 nM T86679 CP02LD 45481765 IC50 > 50000 nM T86679 C0L9GH 45481766 IC50 > 50000 nM T86679 CH54CA 45481767 IC50 > 10000 nM T86679 C7GF4H 45481768 IC50 > 10000 nM T86679 C1FA8U 45481769 IC50 > 10000 nM T86679 C2TWL7 45481770 IC50 > 50000 nM T86679 C5H7SZ 45481771 IC50 = 8630 nM T86679 C12JUY 45482074 IC50 = 50000 nM T86679 C0FG6J 45482075 IC50 = 12400 nM T86679 CQ5ZF6 45482076 IC50 = 13000 nM T86679 CMI3P8 45482077 IC50 > 50000 nM T86679 CDSG82 45482078 IC50 > 10000 nM T86679 C01FXN 45482079 IC50 > 10000 nM T86679 CE3TD2 45482080 IC50 = 5370 nM T86679 C0IT6Y 45482081 IC50 = 1440 nM T86679 C0RN6K 45482082 IC50 = 7370 nM T86679 CD6I4G 45482083 IC50 > 10000 nM T86679 CZ30JX 45482084 IC50 > 50000 nM T86679 CY49LO 45482085 IC50 = 1810 nM T86679 C1VEW8 45482086 IC50 = 906 nM T86679 C8Q6KD 45482087 IC50 = 6450 nM T86679 CP5LN6 45482088 IC50 > 10000 nM T86679 C12UZF 45482089 IC50 > 10000 nM T86679 CIF06H 45482090 IC50 = 1220 nM T86679 CDK76E 45482091 IC50 > 10000 nM T86679 CC52GU 45482092 IC50 > 100000 nM T86679 CL39ZH 45482093 IC50 > 10000 nM T86679 C8PQ9W 45482094 IC50 = 9100 nM T86679 COL2R3 45482462 IC50 > 10000 nM T86679 CNDA49 45482464 IC50 = 5060 nM T86679 C1LM8Y 45486932 Ki = 8130 nM T86679 CPCD97 46175652 IC50 > 50000 nM T86679 CD30NG 46175736 IC50 > 50000 nM T86679 C8GLI6 46175737 IC50 > 50000 nM T86679 C15UPZ 46175738 IC50 > 50000 nM T86679 CQRB27 46175914 IC50 > 50000 nM T86679 CQ9NB4 46176000 IC50 > 50000 nM T86679 CRE07N 46205479 Ki > 10000 nM T86679 C5CV8H 46205480 Ki > 10000 nM T86679 C5GM2E 46205481 Ki > 10000 nM T86679 C7YD4H 46205482 Ki > 10000 nM T86679 C1MS4I 46205483 Ki > 10000 nM T86679 CG60ME 46205484 Ki > 10000 nM T86679 C4B5NU 46205485 Ki > 10000 nM T86679 CQK0G9 46205805 Ki > 10000 nM T86679 CLW1U9 46205806 Ki > 10000 nM T86679 CRS91E 46205807 Ki > 10000 nM T86679 CT8E0B 46205808 Ki > 10000 nM T86679 C5EZ8J 46205809 Ki > 10000 nM T86679 CS3MD6 46205810 Ki > 10000 nM T86679 CLAP45 46206128 Ki > 10000 nM T86679 CK85FB 46206129 Ki > 10000 nM T86679 CTZ2J4 46206130 Ki > 10000 nM T86679 CV1HG3 46206131 Ki > 10000 nM T86679 C0XJ1G 46206132 Ki > 10000 nM T86679 CT4C0Q 46206133 Ki > 10000 nM T86679 C9TY8Z 46206464 Ki > 10000 nM T86679 COIG13 46206465 Ki > 10000 nM T86679 C5NGI1 46206466 Ki > 10000 nM T86679 CYZ9G2 46206467 Ki > 10000 nM T86679 C8JDB5 46206468 Ki > 10000 nM T86679 C45TYC 46206469 Ki > 10000 nM T86679 CHO5B4 46206809 Ki > 10000 nM T86679 CDS62V 46206810 Ki > 10000 nM T86679 C7RP3G 46206811 Ki > 10000 nM T86679 CMIE96 46213946 IC50 = 77 nM T86679 C9E3JO 46227950 Ki = 89.13 nM T86679 CGC6Z1 46227951 Ki = 35.48 nM T86679 C3R1YJ 46227952 Ki = 21.38 nM T86679 C82AHQ 46227957 Ki = 93.33 nM T86679 CFPO49 46227958 Ki = 199.53 nM T86679 CHT97D 46227959 Ki = 61.66 nM T86679 C95RAL 46227973 Ki = 27.54 nM T86679 CFKX20 46227974 Ki = 38.9 nM T86679 CK1A0T 46227980 Ki = 549.54 nM T86679 CHO9J8 46227984 Ki = 32.36 nM T86679 CB83SH 46227993 Ki = 316.23 nM T86679 CP5K0S 46227994 Ki = 162.18 nM T86679 CFGA04 46227995 Ki = 89.13 nM T86679 CUD8P1 46228002 Ki = 125.89 nM T86679 C2MW6U 46228003 Ki = 120.23 nM T86679 C8VE7J 46228004 Ki = 46.77 nM T86679 C4PSD1 46228006 Ki = 12.88 nM T86679 C30RBH 46228011 Ki = 117.49 nM T86679 CMQ4E3 46228016 Ki = 831.76 nM T86679 CM1D4O 46228017 Ki = 645.65 nM T86679 CBV1C2 46228018 Ki = 13.8 nM T86679 CXM4R0 46228022 Ki = 19.05 nM T86679 CE42MY 46228023 Ki = 21.38 nM T86679 CN24EL 46228025 Ki = 275.42 nM T86679 CB5OQ0 46228057 Ki = 269.15 nM T86679 CT61WP 46228058 Ki = 14.79 nM T86679 C5C0LN 46228971 Ki > 1000 nM T86679 C3BVX2 46228972 Ki > 1000 nM T86679 C1HNW9 46228973 Ki > 1000 nM T86679 CBI5E6 46228988 Ki > 1000 nM T86679 C38ZFW 46229140 Ki = 1.39 nM T86679 CAD9G4 46229141 Ki = 4.16 nM T86679 CJ8CU7 46229272 IC50 > 100 nM T86679 C4IN6L 46229273 Ki > 1000 nM T86679 CURG78 46229274 Ki > 1000 nM T86679 CZ9BN5 46229301 Ki > 1000 nM T86679 CEIJ97 46229302 Ki > 1000 nM T86679 CN38YO 46229322 Ki > 1000 nM T86679 C9YX4P 46229323 Ki > 1000 nM T86679 C1KVY2 46230151 EC50 > 10000 nM T86679 C7EWV0 46230238 EC50 > 10000 nM T86679 C80CWB 46230290 EC50 > 10000 nM T86679 CM1H7R 46233161 Ki = 190.55 nM T86679 CW54HP 46233214 Ki = 478.63 nM T86679 CT5CF9 46233315 Ki = 138.04 nM T86679 C8GM6X 46233347 Ki = 371.54 nM T86679 CLK4P1 46233348 Ki = 281.84 nM T86679 C17TOR 46233377 Ki = 35.48 nM T86679 C3MCA6 46233378 Ki = 26.92 nM T86679 C8PJ7D 46233379 Ki = 134.9 nM T86679 C7LY3J 46233380 Ki = 588.84 nM T86679 CG57HC 46237928 IC50 = 49.8 nM T86679 C0Z1AL 46237929 IC50 = 53.9 nM T86679 CB6P5J 46238064 IC50 = 272 nM T86679 CM6K9V 46238066 IC50 = 1327 nM T86679 CMD67R 46238067 IC50 = 1324 nM T86679 C9S4VL 46238068 IC50 = 1467 nM T86679 CO5J9W 46238636 IC50 = 120 nM T86679 CES60L 46238684 IC50 = 145 nM T86679 C5H9JS 46238686 IC50 = 169 nM T86679 CXI4A9 46238694 IC50 = 111 nM T86679 C0I1XV 46238729 IC50 = 172 nM T86679 C3L9OR 46240228 IC50 = 206 nM T86679 CM0O5I 46837562 Ki = 21.88 nM T86679 C72GST 46837563 Ki = 100 nM T86679 CPG0Z6 46837564 Ki = 1047.13 nM T86679 CC7Q8B 46837702 Ki = 114.82 nM T86679 CGN5V6 46837703 Ki = 79.43 nM T86679 CKGM09 46837704 Ki = 2.344 nM T86679 CRG03C 46837705 Ki = 3.548 nM T86679 CX0K7T 46837839 Ki = 30.9 nM T86679 CVD32X 46837841 Ki = 97.72 nM T86679 CT6WJ4 46865897 EC50 = 8870 nM T86679 C5QXL9 46866591 Ki = 1 nM T86679 C8VJ9K 46866592 Ki = 4 nM T86679 CK9AU5 46866593 Ki = 1 nM T86679 CA2S6O 46875997 EC50 > 100000 nM T86679 CY7WL5 46880331 Ki = 380 nM T86679 CL47CE 46880332 Ki = 47 nM T86679 C50XUB 46880372 Ki = 28 nM T86679 CZJ2V5 46880373 Ki = 41 nM T86679 CL8UH3 46880375 Ki = 5 nM T86679 C2P3YO 46880417 Ki = 380 nM T86679 CJ96BI 46880418 Ki = 3668 nM T86679 CQ93IM 46880419 Ki = 5 nM T86679 CMCX40 46880420 Ki = 42 nM T86679 C7P6TS 46880421 Ki = 78 nM T86679 CKB31F 46880422 Ki = 32 nM T86679 CH5B6C 46880424 Ki = 1 nM T86679 CB9TI2 46880470 Ki = 30 nM T86679 C46AYO 46880471 Ki = 134 nM T86679 C0DP5N 46880472 Ki = 202 nM T86679 CSXZ76 46880473 Ki = 72 nM T86679 COQ7X3 46880474 Ki = 2 nM T86679 C2SM9Q 46880475 Ki = 2 nM T86679 CV10FQ 46880506 Ki = 30 nM T86679 CMP72U 46880507 Ki = 4 nM T86679 CM36IE 46880508 Ki = 47 nM T86679 CS2X0C 46880509 Ki = 33 nM T86679 C61JDB 46880510 Ki = 14 nM T86679 C58OJH 46880511 Ki = 208 nM T86679 C1TG8M 46882994 IC50 = 5376 nM T86679 CO0P9H 46882995 IC50 > 10000 nM T86679 C95IFA 46882996 IC50 = 3672 nM T86679 C2F0IA 46882997 IC50 = 758 nM T86679 C14OFC 46882998 IC50 = 1259 nM T86679 C97CLT 46883039 IC50 > 10000 nM T86679 CD50FZ 46883040 IC50 = 5577 nM T86679 CQT47C 46883041 IC50 = 414 nM T86679 CYUD90 46883042 IC50 = 43 nM T86679 CA4O8S 46883043 IC50 = 55 nM T86679 CE12TM 46883070 IC50 = 92 nM T86679 C19PUS 46883071 IC50 = 287 nM T86679 C93JQZ 46883072 IC50 = 944 nM T86679 C5UOJ7 46883073 IC50 = 450 nM T86679 CJG6K1 46883074 IC50 = 4142 nM T86679 CKQG17 46883106 IC50 = 19 nM T86679 C12NEL 46883107 IC50 = 17 nM T86679 CBZ74M 46883108 IC50 = 487 nM T86679 CXQW19 46883109 IC50 = 468 nM T86679 C3T4YP 46883110 IC50 = 18 nM T86679 C4M6IK 46883155 IC50 = 148 nM T86679 CJ1L0R 46883156 IC50 = 176 nM T86679 CD6EW1 46883157 IC50 = 148 nM T86679 CXA5L7 46883158 IC50 = 511 nM T86679 CSK8A5 46883159 IC50 = 215 nM T86679 CS31KC 46883205 IC50 = 1295 nM T86679 CM0Z4K 46883206 IC50 = 109 nM T86679 CG4J3B 46883207 IC50 = 869 nM T86679 CJ57AD 46883208 IC50 = 16 nM T86679 CEV0M1 46885402 EC50 > 100000 nM T86679 C9I6WP 46885403 EC50 > 100000 nM T86679 CFY8H2 46885404 EC50 = 42400 nM T86679 CTYZ06 46885470 EC50 > 100000 nM T86679 C0X4MS 46885471 EC50 = 17100 nM T86679 C28VME 46885472 EC50 = 16800 nM T86679 CCBF03 46885473 EC50 > 100000 nM T86679 C1J2ZP 46885474 EC50 > 100000 nM T86679 CO3AF2 46885516 EC50 > 100000 nM T86679 CUV1X4 46885517 EC50 > 100000 nM T86679 C4A0CV 46885518 EC50 = 20000 nM T86679 CH70LQ 46885547 EC50 > 100000 nM T86679 CVG1D3 46885548 EC50 > 100000 nM T86679 C4TFD0 46885549 EC50 > 100000 nM T86679 C7KD6Q 46885550 EC50 > 100000 nM T86679 C06IZF 46885551 EC50 > 100000 nM T86679 CJ1SV9 46885588 EC50 > 100000 nM T86679 CUFE02 46893147 Ki > 1000 nM T86679 C3JCB1 46911060 Ki = 8 nM T86679 CVT18D 47104774 Ki = 415.7 nM T86679 C02HEX 49797747 Ki = 7 nM T86679 CC61BT 49797748 Ki = 4 nM T86679 C8HA0Y 49797749 Ki = 18 nM T86679 C6XFQ7 49797750 Ki = 23 nM T86679 CP1I3U 49797771 Ki = 8 nM T86679 CN4UQ9 49797772 Ki = 14 nM T86679 CF32QB 49797773 Ki = 4 nM T86679 CB0X1S 49797774 Ki = 22 nM T86679 C21IWV 49797793 Ki = 15 nM T86679 C4Y0JV 49797794 Ki = 10 nM T86679 C6X5LC 49797795 Ki = 19 nM T86679 CD26ZY 49797796 IC50 = 23 nM T86679 CN58DG 49797797 IC50 = 600 nM T86679 CY1XE9 49797825 IC50 = 350 nM T86679 CXJV63 49797826 IC50 = 60 nM T86679 C4JX9B 49797827 IC50 = 6000 nM T86679 CXH10P 49797828 IC50 = 8 nM T86679 CF0H2A 49797852 IC50 = 42 nM T86679 C7SH3X 49797853 IC50 = 77 nM T86679 C7DM9C 49797854 IC50 = 230 nM T86679 CB87EF 49797855 IC50 = 40 nM T86679 CYTS51 49797856 IC50 = 19 nM T86679 C8FD9E 49797878 IC50 = 23 nM T86679 CNRX41 49797879 IC50 = 7 nM T86679 CG2OC1 49797903 IC50 = 21 nM T86679 CU1H3X 49797904 Ki = 19 nM T86679 CO69IE 49797905 Ki = 4 nM T86679 C9AVX7 49797906 Ki = 6 nM T86679 C5R8OV 49798135 Ki = 31.62 nM T86679 CSB23K 49798137 IC50 = 16 nM T86679 CJ15VM 49798138 IC50 = 21 nM T86679 CEC37Y 49798139 Ki = 18 nM T86679 C7P6DN 49798140 Ki = 13 nM T86679 CZIB48 49798161 Ki = 40.74 nM T86679 CJ8CH9 49863226 Ki = 1294 nM T86679 CYKD61 49870828 Ki = 4650 nM T86679 C8WP4Y 49870952 EC50 = 10000 nM T86679 C4WXE2 50925499 Ki = 1.3 nM T86679 C0OQI7 50940921 Ki = 374 nM T86679 C1UMB4 50940926 Ki = 307 nM T86679 CCD60O 50940932 Ki = 3250 nM T86679 CD1U2T 50940964 Ki = 12 nM T86679 CLY1D0 50940966 Ki = 302 nM T86679 CJC06P 50940976 Ki = 1668 nM T86679 CB5TZ6 50940978 Ki = 20.5 nM T86679 C5H8FK 50940980 Ki = 49 nM T86679 CW76LB 50940981 Ki = 164.7 nM T86679 C1B7TN 50941005 Ki = 16.4 nM T86679 C2J0GZ 51039221 IC50 > 10000 nM T86679 CS36WH 51039222 IC50 > 100000 nM T86679 CPY2L4 51039223 IC50 > 10000 nM T86679 CUB5G9 51040798 Ki > 10000 nM T86679 C8P3IT 51050841 IC50 > 10000 nM T86679 COFS19 51050842 IC50 > 30000 nM T86679 C96NLK 51050843 IC50 > 10000 nM T86679 C32PZT 51050844 IC50 = 7140 nM T86679 CYBC20 51050845 IC50 = 20600 nM T86679 CO3N1B 51050939 IC50 > 10000 nM T86679 CGCI34 51050940 IC50 > 10000 nM T86679 C35FWV 51050941 IC50 > 10000 nM T86679 CBX3Q5 51050942 IC50 > 30000 nM T86679 C35OZM 51050943 IC50 > 100000 nM T86679 CRPE85 51050944 IC50 > 100000 nM T86679 CE2ZF4 51051035 IC50 > 100000 nM T86679 C67BTI 51051036 IC50 > 100000 nM T86679 C2WTK7 51051037 IC50 > 100000 nM T86679 CT5Z6U 51051038 IC50 > 100000 nM T86679 C9U0PR 51051039 IC50 > 100000 nM T86679 CG5P0M 51051040 IC50 > 100000 nM T86679 C2F7LS 51051138 IC50 > 100000 nM T86679 C37NQZ 51051140 IC50 = 10700 nM T86679 C72UZF 51051141 IC50 > 30000 nM T86679 CP4Q8Y 51051143 IC50 > 10000 nM T86679 CK12HU 51051145 IC50 > 100000 nM T86679 C6BN9V 51051146 IC50 > 100000 nM T86679 CTZ4H6 51051245 IC50 > 100000 nM T86679 CHX3O5 51051246 IC50 > 100000 nM T86679 CVBO13 51051248 IC50 > 10000 nM T86679 CR2TW4 51051249 IC50 = 11100 nM T86679 C1DB8M 51051251 IC50 = 7060 nM T86679 C7TF3A 51112335 EC50 = 34.67 nM T86679 C8Z0NV 52912216 IC50 > 10000 nM T86679 C8SX6V 52933926 Ki = 560 nM T86679 CT53UX 52941201 Ki = 884 nM T86679 CSGQ69 52941244 Ki = 60 nM T86679 C9H3FM 52941478 IC50 > 50000 nM T86679 C71HWB 52941597 Ki = 3474 nM T86679 C3J6FO 52942359 Ki = 504 nM T86679 CCJP23 52942475 Ki = 2669 nM T86679 CV8EW1 52942501 Ki = 5155 nM T86679 C2BJZ3 52943652 Ki = 1.7 nM T86679 CN10RU 52943791 Ki > 5000 nM T86679 C8NER0 52943888 Ki > 5000 nM T86679 C5I4BV 52944930 Ki = 21 nM T86679 CVB60F 52945006 Ki > 5000 nM T86679 C2H9AY 52945064 Ki = 3655 nM T86679 CJAY05 52945098 Ki = 70 nM T86679 C45SQC 52945195 Ki = 0.44 nM T86679 CHT4Z6 52946113 Ki = 17 nM T86679 CX9G3T 52946114 Ki = 70 nM T86679 CK76UG 52946159 Ki = 291 nM T86679 CEFW97 52946211 IC50 > 50000 nM T86679 CUA1O9 52946453 Ki = 1 nM T86679 C28VAP 52947301 Ki = 187 nM T86679 C7HY0V 52947452 Ki = 172 nM T86679 CV9D1Y 52947525 IC50 = 1100 nM T86679 C4KA6Y 52948671 Ki = 633 nM T86679 COW0J3 52948763 Ki > 5000 nM T86679 C3B9OG 52948788 IC50 = 19000 nM T86679 C7TI2R 52948915 Ki = 10 nM T86679 C28MQF 52948949 Ki = 19 nM T86679 CQ91YN 52948995 IC50 > 50000 nM T86679 CE8F3G 52949755 Ki = 1933 nM T86679 CE3XQ7 52949772 Ki > 10000 nM T86679 CL6K9M 52949999 Ki = 710 nM T86679 C74BRO 52950000 Ki = 338 nM T86679 CHM1G6 52950027 Ki = 330 nM T86679 C0L8VT 52950028 Ki = 3413 nM T86679 CQAP62 52950040 Ki = 0.4 nM T86679 C3JEO8 52950206 Ki = 1675 nM T86679 CRB59S 53242165 IC50 = 20 nM T86679 CI35WL 53248698 IC50 = 14 nM T86679 CDS80Q 53248700 Ki = 5 nM T86679 CJZ98W 53318744 Ki = 13 nM T86679 C5F1IR 53318745 Ki = 2 nM T86679 C5HL4R 53321372 Ki = 26 nM T86679 CA91KC 53322692 Ki = 6 nM T86679 CH7O8A 53324032 Ki = 0.6 nM T86679 CY04CM 53325341 Ki = 43 nM T86679 CH6X9F 53354632 Ki = 39.81 nM T86679 CUO97T 54577823 Ki = 12500 nM T86679 CZQ2H9 54580150 IC50 = 44 nM T86679 C9LU8J 54580623 Ki > 30000 nM T86679 C84FJX 54581142 IC50 = 13 nM T86679 CSX07T 54581143 IC50 = 8 nM T86679 C85ZXD 54582166 IC50 = 8 nM T86679 C2C8MB 54582167 Ki = 18 nM T86679 CHDV60 54583133 IC50 = 19 nM T86679 CS6O9E 54584124 IC50 = 17 nM T86679 C7CWY9 54584125 IC50 = 49 nM T86679 C3N7RC 54585057 IC50 = 26 nM T86679 CO7IC0 54585058 IC50 = 18 nM T86679 CKCD81 54585511 Ki > 30000 nM T86679 C02CVB 54586036 IC50 = 41 nM T86679 C6IV3L 54587015 IC50 = 42 nM T86679 CTFS79 54587016 IC50 = 72 nM T86679 CSL08D 54587662 Ki > 30000 nM T86679 C83VFS 54754508 Ki > 10000 nM T86679 C40IVD 54768079 Ki > 10000 nM T86679 C1UW4E 54768080 Ki > 10000 nM T86679 C4JA9T 54768112 Ki > 10000 nM T86679 C2JPC3 54768115 Ki > 10000 nM T86679 CL5SE3 54768601 Ki > 10000 nM T86679 C6SYD1 54768602 Ki = 800 nM T86679 CX9A4R 54768635 Ki > 10000 nM T86679 C3HNS6 54768636 Ki > 10000 nM T86679 CB7T1O 56627882 EC50 = 542 nM T86679 C6WSF9 56657920 Ki > 10000 nM T86679 CD7C2P 56661442 Ki > 30000 nM T86679 C2FI4U 56661443 Ki > 10000 nM T86679 CVLM74 56664888 Ki > 10000 nM T86679 CBQS24 56668308 Ki > 30000 nM T86679 CYNJ53 56668410 Ki > 10000 nM T86679 CWM34N 56668411 Ki > 10000 nM T86679 CSJ34D 56668412 Ki > 10000 nM T86679 C98FPH 56671922 Ki > 10000 nM T86679 CD6C0P 56675199 Ki > 10000 nM T86679 CH8YR5 56675200 Ki > 30000 nM T86679 CUJ34X 56675201 Ki > 30000 nM T86679 CK3AZ9 56675297 Ki > 10000 nM T86679 C58FTQ 56675298 Ki > 10000 nM T86679 C7TNW9 56675299 Ki > 10000 nM T86679 CDN69Q 56678498 Ki > 10000 nM T86679 C13UZX 56678638 Ki > 10000 nM T86679 CM04LK 56678639 Ki > 10000 nM T86679 CVP0A9 56681843 Ki > 10000 nM T86679 CPQL51 56783276 EC50 = 34.67 nM T86679 C02DIY 56838950 Ki > 10000 nM T86679 CYS17U 56844240 Ki = 50.12 nM T86679 COY13J 56924646 Ki = 4 nM T86679 CH1JR4 56950235 IC50 = 838 nM T86679 CXB8Z6 56951623 Ki = 7.5 nM T86679 C9T1XQ 56964459 IC50 = 2.42 nM T86679 CY1IG3 56964460 IC50 = 2.11 nM T86679 CZ42XV 56964461 IC50 = 2.5 nM T86679 CC50SG 56964576 IC50 = 3.1 nM T86679 CHR8L5 57325914 IC50 = 5.34 nM T86679 C7SRT3 57325915 IC50 = 7850 nM T86679 CREU79 57328471 IC50 > 30000 nM T86679 C8JY3E 57384287 EC50 = 1489 nM T86679 CYSA75 57384288 EC50 = 6069 nM T86679 CDN54M 57384289 EC50 = 739 nM T86679 CA63RT 57384543 EC50 = 2279 nM T86679 CW63IC 57384544 EC50 = 40310 nM T86679 CCPY02 57385043 EC50 = 12160 nM T86679 CKO3L1 57387337 EC50 = 2.3 nM T86679 C8X7MO 57387594 EC50 = 14 nM T86679 C6XKL9 57387596 EC50 = 120 nM T86679 C7XW0T 57387822 EC50 = 6694 nM T86679 CT1R6Q 57387824 EC50 = 126 nM T86679 C01AHY 57387825 EC50 = 355 nM T86679 CNL3P2 57388054 EC50 = 1173 nM T86679 CK7R6O 57388055 EC50 = 257 nM T86679 CMBN74 57388056 EC50 = 296 nM T86679 C1BAX6 57391653 IC50 = 251 nM T86679 C45GCN 57391694 IC50 = 319 nM T86679 C03HUE 57391695 IC50 = 915 nM T86679 CJF61Z 57391696 IC50 > 1000 nM T86679 CC3X7G 57393433 IC50 = 772 nM T86679 C1B3QM 57393434 IC50 > 1000 nM T86679 C8ZX4L 57393435 IC50 > 1000 nM T86679 CVO2P8 57395120 IC50 = 906 nM T86679 C9VWH7 57395161 IC50 > 1000 nM T86679 CJM7E8 57395162 IC50 = 595 nM T86679 CEQR05 57395163 IC50 = 122 nM T86679 CDP13M 57395164 IC50 = 580 nM T86679 CSTG21 57396888 IC50 = 46 nM T86679 CWX64M 57396935 IC50 = 31 nM T86679 CC52TB 57396936 IC50 = 45 nM T86679 C1WT0H 57396937 IC50 > 1000 nM T86679 CD6JT5 57398641 IC50 = 90 nM T86679 CHC8U6 57398676 IC50 = 32 nM T86679 C1J3DG 57400352 IC50 = 40 nM T86679 CNRY34 57400353 IC50 = 863 nM T86679 CIX58U 57402117 IC50 = 42 nM T86679 CLCX61 57402118 IC50 = 740 nM T86679 CBMP08 57402160 IC50 > 1000 nM T86679 C58APE 57402161 IC50 = 33 nM T86679 CKB51R 57402162 IC50 = 548 nM T86679 CQK46U 57402163 IC50 > 1000 nM T86679 CYHD10 57403904 IC50 = 32 nM T86679 CD2NO5 57403905 IC50 = 27 nM T86679 C5HF9M 57429602 Ki = 3.6 nM T86679 C9GB1E 57429603 Ki = 4.9 nM T86679 CGU5V6 57429605 Ki = 3.5 nM T86679 C0EI8F 57429607 Ki = 3.7 nM T86679 CLCR39 57429608 Ki = 12 nM T86679 CU9LK1 57429610 Ki = 9.9 nM T86679 CUG3Y7 57429611 Ki = 130 nM T86679 C4SH9E 57429615 Ki = 2.2 nM T86679 CRC4W0 57429616 Ki = 2.8 nM T86679 C50EVU 57429617 Ki = 1.6 nM T86679 C8M1JK 57429618 Ki = 3 nM T86679 C50JLY 57429619 Ki = 1.3 nM T86679 CXZ53C 57429620 Ki = 1.6 nM T86679 C49JKZ 57429621 Ki = 48 nM T86679 CT1PH5 57429644 Ki = 2.6 nM T86679 C9R5GB 57429645 Ki = 4 nM T86679 C54JLY 57429647 Ki = 1.2 nM T86679 C05DRY 57429649 Ki = 1.5 nM T86679 CPZ25B 57429658 Ki > 600 nM T86679 CA7O2M 57429661 Ki = 6 nM T86679 CC2EI5 57988776 Ki = 5.4 nM T86679 CPT7K6 57988777 Ki = 3.6 nM T86679 C35CPN 57988794 Ki = 62 nM T86679 C1HU4O 59011969 Ki > 10000 nM T86679 C7NW3Q 59351824 IC50 = 480 nM T86679 C5G2RH 60154738 IC50 = 505 nM T86679 C4U7BI 60154739 IC50 = 2122 nM T86679 CU3R2Q 60154740 IC50 = 3244 nM T86679 CJ57XU 60154742 IC50 = 3235 nM T86679 CUK15D 60154835 IC50 = 2144 nM T86679 CK7VH4 60154837 IC50 > 5000 nM T86679 C3PO4T 60155712 IC50 = 2428 nM T86679 CJB03P 60155713 IC50 > 5000 nM T86679 C6W8XE 60155714 IC50 > 5000 nM T86679 CN03ZC 60155715 IC50 > 5000 nM T86679 CEZ4V5 60155716 IC50 > 5000 nM T86679 C1ZXO7 60155796 IC50 = 2061 nM T86679 CZRU45 60155797 IC50 > 5000 nM T86679 C8GZ3V 60155798 IC50 > 5000 nM T86679 CXLO10 60155799 IC50 > 5000 nM T86679 CYB1L4 60155893 IC50 > 5000 nM T86679 C0B5OZ 60155894 IC50 > 5000 nM T86679 CB9A6F 60155895 IC50 > 5000 nM T86679 C2VPM8 60155896 IC50 > 5000 nM T86679 CW7R1L 60155897 IC50 > 5000 nM T86679 CP3H2Z 60156002 IC50 > 5000 nM T86679 C8KU5V 60156003 IC50 > 5000 nM T86679 C2LN4J 60156004 IC50 > 5000 nM T86679 C8SZE0 60156005 IC50 > 5000 nM T86679 CGL84Y 60156006 IC50 > 5000 nM T86679 CFBG07 60156104 IC50 > 5000 nM T86679 CKVJ21 60156105 IC50 = 1107 nM T86679 C7L1BF 60156106 IC50 = 1755 nM T86679 C38NUA 60156107 IC50 = 1542 nM T86679 C87SMR 60156108 IC50 = 1042 nM T86679 C20XJH 66892244 Ki = 14 nM T86679 CWN0X9 66892382 Ki = 6 nM T86679 CD37KG 66892501 Ki = 23 nM T86679 CH91RG 66892710 Ki = 12 nM T86679 CV6PW1 66892867 Ki = 4 nM T86679 C8GXZ4 66892978 Ki = 77 nM T86679 CCA5E2 66893166 Ki = 9.7 nM T86679 C4TCU3 66893508 Ki = 21.6 nM T86679 CDIC80 66893509 Ki = 4 nM T86679 CY1FM6 66893874 Ki = 6.5 nM T86679 CEK1C2 66894029 Ki = 8.7 nM T86679 CBL0Y1 66894035 Ki = 9 nM T86679 C0RPT4 66894039 Ki = 17.5 nM T86679 CK4BU2 66894080 Ki = 24 nM T86679 CP4LZ8 66894103 Ki = 7.5 nM T86679 CR93KL 66894143 Ki = 9 nM T86679 C9GDP5 66894241 Ki = 0.9 nM T86679 CGK4F8 66894243 Ki = 41 nM T86679 CHE2D4 66894271 Ki = 43 nM T86679 C20XUT 66894327 Ki = 9 nM T86679 C4WC7I 66894703 Ki = 19 nM T86679 CND2X4 66899873 Ki = 1 nM T86679 C1XZV9 67364057 Ki = 158.49 nM T86679 CW37UH 67548131 IC50 = 368 nM T86679 C56UIN 67548175 IC50 = 146 nM T86679 C6VKP4 67548337 IC50 = 459 nM T86679 CGXY26 67548392 IC50 = 94 nM T86679 C5U3WL 67548498 IC50 > 1000 nM T86679 CC4Y6V 67548720 IC50 = 263 nM T86679 C8B1JS 67548983 IC50 > 1000 nM T86679 CPQ2I7 67549056 IC50 > 1000 nM T86679 C71HZU 67549086 IC50 = 90 nM T86679 C74YXW 67549097 IC50 > 1000 nM T86679 CD09WI 67549451 IC50 > 1000 nM T86679 C5M0NT 67549626 IC50 > 1000 nM T86679 C8Z7RX 67549879 IC50 = 95 nM T86679 C18CNK 68405754 IC50 > 1000 nM T86679 CNYS04 68405874 IC50 > 1000 nM T86679 CWEQ54 68405927 IC50 > 268 nM T86679 CA12YE 69028196 Ki = 13 nM T86679 C2OM6I 69029783 Ki = 3 nM T86679 CIL82V 69029798 Ki = 4 nM T86679 CQK0D8 69030381 Ki = 4.5 nM T86679 CU7IZ5 69030489 Ki = 8 nM T86679 CVBE74 69030712 Ki = 10.7 nM T86679 CWPZ35 69031242 Ki = 4.6 nM T86679 CRL75S 69031481 Ki = 4 nM T86679 CU5N7K 69031810 Ki = 14 nM T86679 C2WLR9 69032552 Ki = 13.7 nM T86679 C0P1OR 69427076 EC50 = 2700 nM T86679 CXUB67 69846372 Ki > 10000 nM T86679 C76KTS 69846756 Ki > 30000 nM T86679 CCDH27 69961639 EC50 = 885 nM T86679 CS0I7Z 70682890 EC50 = 1700 nM T86679 C7LZO2 70683991 Ki = 10000 nM T86679 CN86WI 70686119 Ki = 1000 nM T86679 CB3D6N 70688247 Ki = 10000 nM T86679 C1KJD5 70689262 EC50 = 2000 nM T86679 C8XWN2 70696536 Ki = 630.96 nM T86679 C2EW3D 70696537 Ki = 1258.93 nM T86679 C7USK0 70696572 Ki > 10000 nM T86679 CBN9A8 70697521 EC50 = 6100 nM T86679 C75JTG 71361867 Ki > 30000 nM T86679 C31FGM 71412032 Ki = 140 nM T86679 CBZM95 71449068 EC50 > 10000 nM T86679 CXZ40U 71450227 Ki > 10000 nM T86679 C38UKP 71450240 Ki > 10000 nM T86679 CXM83Y 71450241 Ki = 2110 nM T86679 C9G0FP 71450242 Ki = 6590 nM T86679 CC73UY 71450243 Ki > 10000 nM T86679 CW75JC 71450849 EC50 > 10000 nM T86679 C4VMP7 71451329 Ki = 1540 nM T86679 C4LVT1 71452054 Ki > 10000 nM T86679 CC2Q9H 71452055 Ki > 10000 nM T86679 CQ4CA3 71452056 Ki = 5290 nM T86679 CWOB13 71452072 Ki = 7660 nM T86679 C0MD9G 71452718 Ki = 5.3 nM T86679 C0NC4G 71453140 Ki > 10000 nM T86679 C9QD3W 71453871 Ki > 10000 nM T86679 CKW2G6 71453872 Ki > 10000 nM T86679 C0VK4E 71453873 Ki > 10000 nM T86679 CR8A0V 71453874 Ki = 3330 nM T86679 CV0NW6 71453875 Ki > 3000 nM T86679 C5S3FU 71453891 Ki = 9300 nM T86679 C0M9CP 71453892 Ki = 2160 nM T86679 CY1B4N 71453893 Ki > 10000 nM T86679 C76PJS 71453894 Ki = 6320 nM T86679 C56VEI 71455599 Ki > 10000 nM T86679 C79IVN 71455600 Ki > 10000 nM T86679 CM2ZF9 71455601 Ki = 7500 nM T86679 CEO64T 71455602 Ki > 10000 nM T86679 CPN0B7 71455603 Ki = 3940 nM T86679 CUE71P 71455604 Ki = 9840 nM T86679 CC1RD4 71455619 Ki = 3880 nM T86679 C2ITP7 71455620 Ki = 5260 nM T86679 CQ8U5S 71455621 Ki = 4810 nM T86679 CB2E9C 71455622 Ki = 3980 nM T86679 CTH1W7 71455623 Ki > 10000 nM T86679 C1QLP9 71455624 Ki = 1110 nM T86679 CVJZ12 71456194 EC50 >= 10000 nM T86679 CJBC05 71456195 EC50 >= 10000 nM T86679 CKU1O4 71456259 EC50 = 30000 nM T86679 C5BHA3 71457388 Ki > 10000 nM T86679 CYTZ37 71457389 Ki = 8500 nM T86679 C3H2QF 71457390 Ki = 12200 nM T86679 CPBO67 71457391 Ki = 2620 nM T86679 C12PEI 71457403 Ki = 7470 nM T86679 C19MUP 71457404 Ki = 9720 nM T86679 CS6Z4N 71457405 Ki = 3860 nM T86679 C5RD0O 71457406 Ki > 10000 nM T86679 C6MF5O 71457407 Ki = 2650 nM T86679 CU0YQ6 71459244 Ki > 10000 nM T86679 CV3L0D 71459245 Ki > 10000 nM T86679 CDW92B 71459246 Ki > 10000 nM T86679 C5WX8S 71459247 Ki > 10000 nM T86679 CN79LY 71459248 Ki > 10000 nM T86679 C82QUK 71459249 Ki > 10000 nM T86679 CC9I6G 71459250 Ki > 3000 nM T86679 CQ7BP5 71459268 Ki = 2870 nM T86679 CUI7X3 71459958 EC50 = 13000 nM T86679 C8AY0D 71460344 Ki > 10000 nM T86679 CB9A8S 71461026 Ki > 10000 nM T86679 C60OEP 71461027 Ki > 10000 nM T86679 CUDN57 71461028 Ki = 3180 nM T86679 CJ9K0H 71461029 Ki > 10000 nM T86679 CDX9O4 71461045 Ki > 10000 nM T86679 CA0EJ2 71462751 Ki > 10000 nM T86679 CK7OB3 71462752 Ki > 3000 nM T86679 CP07FL 71462753 Ki > 10000 nM T86679 CK97MP 71462754 Ki > 10000 nM T86679 CV1QN8 71462755 Ki = 2790 nM T86679 COU6E4 71462772 Ki > 10000 nM T86679 CGC23V 71462773 Ki = 2600 nM T86679 C1HAS6 71462774 Ki = 1750 nM T86679 CHT04N 71462775 Ki = 9650 nM T86679 CGT9W5 71508481 IC50 = 120 nM T86679 C79QVF 71508699 Ki > 10000 nM T86679 CLDQ30 71508726 Ki > 10000 nM T86679 CNKZ09 71528098 IC50 > 30000 nM T86679 CT29GM 71570217 Ki = 67.5 nM T86679 CKGR23 71570366 Ki = 493.7 nM T86679 CI39JB 71601630 IC50 = 320 nM T86679 C9J4OB 71601631 IC50 = 440 nM T86679 CRQP84 71601632 IC50 = 420 nM T86679 CNZ17D 71657835 EC50 = 95.5 nM T86679 C70SIG 71680729 Ki > 1000 nM T86679 C0YW1C 71680730 Ki = 679 nM T86679 CG6EY1 71680731 Ki > 1000 nM T86679 CN0WU1 71680732 Ki > 1000 nM T86679 CK2Y6A 71680733 Ki > 1000 nM T86679 CH5KU9 71680734 Ki = 302 nM T86679 C6OXR9 71680735 Ki >= 1000 nM T86679 CA50LT 71680889 Ki > 1000 nM T86679 CCM92I 71680890 Ki = 119 nM T86679 CS51FY 71680891 Ki >= 1000 nM T86679 CX4BZ6 71680892 Ki > 1000 nM T86679 CC7MA1 71680893 Ki > 1000 nM T86679 C6HZ4O 71680894 Ki > 1000 nM T86679 CN0EZ6 71680895 Ki > 1000 nM T86679 C30NCG 71681049 Ki > 1000 nM T86679 C2TR7P 71681050 Ki > 1000 nM T86679 CVY85K 71681051 Ki = 408 nM T86679 C8TCR6 71681052 Ki > 1000 nM T86679 C4KB8W 71681053 Ki > 1000 nM T86679 CLBD58 71681054 Ki > 1000 nM T86679 C50TBU 71681055 Ki = 547 nM T86679 C2Y3KO 71681203 Ki = 361 nM T86679 CIM0S3 71681204 Ki > 1000 nM T86679 C21UWV 71683091 Ki = 365 nM T86679 COWX82 71683092 Ki = 225 nM T86679 C9CLQ3 71683093 Ki > 1000 nM T86679 CV5O0H 71683094 Ki = 801 nM T86679 CCJ17F 71683095 Ki > 1000 nM T86679 C3RD0E 71713167 Ki > 30000 nM T86679 C5NHJ0 72141742 EC50 = 16.98 nM T86679 C5EMX3 72197342 Ki > 10000 nM T86679 C4E0QC 72197343 Ki > 10000 nM T86679 C76ASV 72197513 Ki > 30000 nM T86679 CZW4Y0 72197514 Ki > 10000 nM T86679 CUL8V0 72197515 Ki > 10000 nM T86679 CXF4U1 72197516 Ki > 10000 nM T86679 C3QYT8 72197517 Ki > 10000 nM T86679 C4W8LQ 72197698 Ki > 10000 nM T86679 CY8GU4 72197699 Ki > 10000 nM T86679 C6BUC3 72197700 Ki > 10000 nM T86679 C48QTY 72197701 Ki = 9110 nM T86679 C4D8WO 72197702 Ki > 10000 nM T86679 CAY6J2 72197703 Ki = 841 nM T86679 C6RDT4 72197880 Ki = 2.78 nM T86679 C7XN0S 72197881 Ki > 10000 nM T86679 C5J9QH 72197882 Ki > 10000 nM T86679 CB05ET 72197883 Ki = 8000 nM T86679 C52QMK 72197884 Ki > 10000 nM T86679 CVY9E5 72546298 Ki = 714.6 nM T86679 CGY90F 72546539 Ki = 256.1 nM T86679 C6RPM0 72546540 Ki = 3428 nM T86679 CS81LQ 72696144 Ki > 1000 nM T86679 C3BEM8 72696145 Ki > 1000 nM T86679 C1E4ZD 72696146 Ki > 1000 nM T86679 CQ35NL 72696147 Ki > 1000 nM T86679 CRN4B1 72696148 Ki > 1000 nM T86679 C0IF1J 72696149 Ki > 1000 nM T86679 CL2H7Y 72696273 Ki > 1000 nM T86679 C7MX9Y 72696274 Ki > 1000 nM T86679 CBTE63 72696275 Ki > 1000 nM T86679 CPI89R 72696276 Ki > 1000 nM T86679 COX4B1 72696277 Ki > 1000 nM T86679 CI9HP7 72696397 Ki > 1000 nM T86679 C1RFY6 72696398 Ki > 1000 nM T86679 CY56RG 72696399 Ki > 1000 nM T86679 C6A8ZF 72696400 Ki > 1000 nM T86679 C8ARZ1 72696401 Ki > 1000 nM T86679 CQ4JZ3 72696520 Ki > 1000 nM T86679 C4DN3V 72696521 Ki > 1000 nM T86679 CWG0U4 72697647 Ki > 1000 nM T86679 CH90JS 72697648 Ki > 1000 nM T86679 CPB7K4 72697649 Ki = 3860 nM T86679 C1D7VQ 72697650 Ki > 1000 nM T86679 C81TXZ 72697651 Ki > 1000 nM T86679 CA5BI1 72697652 Ki = 3520 nM T86679 C50SYX 72697785 Ki > 1000 nM T86679 CXPB58 72697786 Ki > 1000 nM T86679 CJ5W1R 72697787 Ki > 1000 nM T86679 C0CJ6R 72697788 Ki > 300 nM T86679 CY1I8G 72697789 Ki = 1740 nM T86679 CXDT98 72697790 Ki > 1000 nM T86679 CS7VK8 72697791 Ki > 10000 nM T86679 CX69MI 72697928 Ki > 1000 nM T86679 CT2L7J 72697929 Ki > 1000 nM T86679 CEWO96 72697930 Ki > 1000 nM T86679 CNP9S3 72697931 Ki = 3970 nM T86679 C3NR4V 72697932 Ki = 17100 nM T86679 CQ4IE7 72697933 Ki > 1000 nM T86679 CY94KO 72697934 Ki > 1000 nM T86679 CO5K1Y 72698079 Ki > 1000 nM T86679 CVB0Y9 72698080 Ki > 1000 nM T86679 CCOP98 72698081 Ki > 1000 nM T86679 C50ZUX 72698082 Ki > 1000 nM T86679 CZG6V9 72698083 Ki > 1000 nM T86679 C97FMG 72698084 Ki > 1000 nM T86679 CH6Z2U 72698223 Ki > 1000 nM T86679 C3QVP5 72698224 Ki > 1000 nM T86679 CBD03K 72698225 Ki > 1000 nM T86679 CST61L 72698226 Ki > 1000 nM T86679 CJ0GB6 72698227 Ki > 300 nM T86679 CKP9M2 72698228 Ki > 1000 nM T86679 CTJ0U3 73348946 Ki > 10000 nM T86679 CI65VU 73349920 EC50 >= 10000 nM T86679 C4C0GK 73349930 EC50 >= 10000 nM T86679 CY2PU1 74944536 IC50 = 1.06 nM T86679 CMS65T 76309882 Ki = 792 nM T86679 CB84HP 76309883 Ki > 30000 nM T86679 C02EBL 76309925 Ki > 10000 nM T86679 C8I4OH 76309932 Ki = 3111 nM T86679 CYHX45 76309933 Ki = 1151 nM T86679 CX1H6Y 76310493 Ki > 10000 nM T86679 C9DL1B 76310832 Ki = 1.97 nM T86679 CCX8V6 76311194 EC50 = 158.49 nM T86679 CQLE57 76311197 EC50 = 1258.93 nM T86679 CSV43U 76313599 Ki > 30000 nM T86679 CP2TA1 76313600 Ki = 5070 nM T86679 CQ5Z4P 76313639 Ki > 10000 nM T86679 CY8D4J 76313640 Ki > 10000 nM T86679 CB0WN9 76313641 Ki > 10000 nM T86679 CNBZ82 76313652 Ki = 194.2 nM T86679 C1C3LK 76314155 Ki > 20000 nM T86679 C25LDC 76314450 Ki = 4.95 nM T86679 CZX45G 76314797 EC50 > 10000 nM T86679 C21BCT 76317721 Ki > 20000 nM T86679 C2K6XR 76317722 Ki > 20000 nM T86679 CY3V7H 76317723 Ki > 20000 nM T86679 CXQY23 76317724 Ki > 20000 nM T86679 CCY8V2 76318040 Ki = 2.9 nM T86679 CL4JH8 76318403 EC50 = 199.53 nM T86679 C9O4CQ 76320863 Ki > 10000 nM T86679 C26VRI 76320870 Ki = 1486 nM T86679 CKLB89 76320909 Ki = 187 nM T86679 CL46PW 76321429 Ki > 20000 nM T86679 CWO42D 76321430 Ki > 10000 nM T86679 CFN3M9 76321431 Ki > 20000 nM T86679 CY5TN2 76321753 Ki = 2.59 nM T86679 C5R6OT 76322076 EC50 = 199.53 nM T86679 CK5Z6L 76324475 Ki = 6250 nM T86679 CHWO53 76324476 Ki = 786 nM T86679 C3CE4B 76324522 Ki > 10000 nM T86679 C9IL0H 76324530 Ki = 43.1 nM T86679 C6AV9Z 76325026 Ki > 20000 nM T86679 C1JV7S 76325027 Ki > 20000 nM T86679 CQ51JN 76325369 Ki = 1.34 nM T86679 C2DPT3 76325370 Ki > 10 nM T86679 CP4CY1 76325371 Ki = 1.05 nM T86679 C5J4ML 76325372 Ki > 10 nM T86679 COD78V 76325693 EC50 > 10000 nM T86679 C3FE0S 76325694 EC50 = 2511.89 nM T86679 CC67KO 76328082 Ki > 10000 nM T86679 CA0MJ2 76328083 Ki > 10000 nM T86679 C72UFI 76328084 Ki > 10000 nM T86679 CNM0E1 76328596 Ki > 20000 nM T86679 CXTN91 76328597 Ki > 20000 nM T86679 C3TH4J 76328598 Ki > 20000 nM T86679 CQI9X5 76328599 Ki > 20000 nM T86679 C0AE9L 76328600 Ki > 20000 nM T86679 C5B0UO 76328910 Ki = 0.17 nM T86679 C5VEJ9 76328911 Ki > 10 nM T86679 C8O5KF 76329263 EC50 = 158.49 nM T86679 C9O0UH 76329264 EC50 > 10000 nM T86679 CF82DA 76329265 EC50 = 794.33 nM T86679 CPVN52 76329266 EC50 = 125.89 nM T86679 CG30CO 76331702 Ki = 250 nM T86679 C6QY2P 76331703 Ki = 2780 nM T86679 CFNG34 76331754 Ki > 10000 nM T86679 CMR14L 76331755 Ki > 10000 nM T86679 CR74DH 76331767 Ki = 4259 nM T86679 CQT81A 76332277 Ki > 20000 nM T86679 CH64XC 76332278 Ki > 20000 nM T86679 CQWD47 76332279 Ki > 20000 nM T86679 CJKD34 76332280 Ki > 20000 nM T86679 C1GZ8R 76332281 Ki > 20000 nM T86679 CVT1E3 76332599 Ki > 10 nM T86679 CVS3F8 76332600 Ki > 10 nM T86679 CYK39X 76332918 EC50 > 10000 nM T86679 C4S8NF 76332919 EC50 = 1584.89 nM T86679 CF68KC 76335303 Ki = 350 nM T86679 CL83MV 76335304 Ki = 2510 nM T86679 C7KY5A 76335305 Ki = 470 nM T86679 CC5IO4 76335344 Ki > 10000 nM T86679 C7FE5D 76335345 Ki > 10000 nM T86679 CIT36F 76335346 Ki > 10000 nM T86679 CV05FX 76335917 Ki > 10000 nM T86679 CLN8S6 76335918 Ki > 20000 nM T86679 CM0D3G 76335919 Ki > 20000 nM T86679 CO86UR 76335920 Ki >= 10000 nM T86679 CESR09 76335921 Ki > 10000 nM T86679 CR85PG 76335922 Ki > 20000 nM T86679 C3HE2N 76335923 Ki > 10000 nM T86679 C5DSC0 76335924 Ki > 20000 nM T86679 C5VM4Q 76336198 Ki = 1 nM T86679 CH9WJ4 76336525 EC50 = 1584.89 nM T86679 CNL62P 76336526 EC50 = 5011.87 nM T86679 C5ZRE9 76336527 EC50 = 398.11 nM T86679 CFWX23 82018566 Ki > 1000 nM T86679 CI4M9P 85706712 Ki > 30000 nM T86679 CGAL51 89534951 EC50 = 94 nM T86679 CB51WQ 90654601 Ki = 42 nM T86679 C0ROS7 101874280 Ki = 2450 nM T86679 CGBO72 118016229 IC50 = 59 nM T86679 C2LIQ1 118016325 IC50 = 2100 nM T86679 CFH85E 118707843 Ki > 30000 nM T86679 COX73K 118707844 Ki = 5320 nM T86679 CR13GS 118707845 Ki = 1180 nM T86679 CS0WC2 118707846 Ki > 30000 nM T86679 C2A3FW 118707847 Ki = 4840 nM T86679 CJ58XH 118707848 Ki > 30000 nM T86679 CF78CL 118707849 Ki > 30000 nM T86679 C3K7UV 118707850 Ki > 30000 nM T86679 C0UFO4 118707851 Ki = 1900 nM T86679 CSW70B 118707852 Ki > 30000 nM T86679 CU9OE7 118707853 Ki > 30000 nM T86679 CGJW82 118707854 Ki > 30000 nM T86679 CUR32J 118707855 Ki = 3060 nM T86679 C6O0RY 118707856 Ki > 10000 nM T86679 CG10IH 118707857 Ki = 10000 nM T86679 C9OHF2 118707858 Ki > 10000 nM T86679 CW72CL 118707859 Ki = 2260 nM T86679 CL0U3C 118707860 Ki = 4620 nM T86679 CL3NG5 118707861 Ki > 10000 nM T86679 C9BSD0 118707862 Ki = 2510 nM T86679 CDTJ73 118707863 Ki = 10000 nM T86679 CRDU39 118707864 Ki = 4810 nM T86679 C6Y5VQ 118707865 Ki = 1970 nM T86679 CBO8V9 118707866 Ki = 1630 nM T86679 C4CU6D 118707867 Ki = 2040 nM T86679 C4P5GH 118707868 Ki > 30000 nM T86679 C9FKE5 118707869 Ki > 30000 nM T86679 CNJ3Z4 118707870 Ki > 3000 nM T86679 CXQY36 118707871 Ki > 10000 nM T86679 C7SL4C 118707872 Ki > 10000 nM T86679 CFR3Z1 118707873 Ki > 10000 nM T86679 C87ATB 118707874 Ki > 10000 nM T86679 C7HS6T 118707875 Ki > 10000 nM T86679 CXHQ82 118707876 Ki > 10000 nM T86679 CEQP75 118707877 Ki > 10000 nM T86679 CY8OV1 118707878 Ki > 10000 nM T86679 CH5B6Y 118707879 Ki = 7150 nM T86679 C3OJW0 118707880 Ki > 10000 nM T86679 CM5BE7 118707881 Ki > 10000 nM T86679 CHR1E9 118707882 Ki > 10000 nM T86679 CZW6U4 118707883 Ki > 10000 nM T86679 COR57B 118707884 Ki > 10000 nM T86679 C8C9TQ 118707885 Ki > 10000 nM T86679 C0NQ2O 118707886 Ki > 10000 nM T86679 CG68RH 118707887 Ki > 10000 nM T86679 C9CY3P 118707888 Ki > 10000 nM T86679 CNC81J 118707889 Ki > 10000 nM T86679 CM53PE 118707890 Ki > 10000 nM T86679 CL4B7K 118707891 Ki > 30000 nM T86679 CR20MO 118707892 Ki > 30000 nM T86679 C8WQ5E 118707893 Ki > 30000 nM T86679 CI6O9D 118707894 Ki > 30000 nM T86679 C28ABD 118707895 Ki > 30000 nM T86679 C56KNQ 118707896 Ki > 30000 nM T86679 C74OYF 118708214 IC50 = 630 nM T86679 CFOC02 118708225 IC50 = 123 nM T86679 CWU94Y 118708234 IC50 = 432 nM T86679 CI29WS 118708235 IC50 = 387 nM T86679 C2B0KW 118708236 IC50 = 334 nM T86679 CX2B8P 118708238 IC50 = 247 nM T86679 CQWJ06 118708239 IC50 = 314 nM T86679 CI76CX 118719026 EC50 = 6100 nM T86679 CM3S0N 118732278 Ki > 20000 nM T86679 CWQ54J 118732279 Ki > 20000 nM T86679 CQL0K7 118732280 Ki > 20000 nM T86679 CRK7H9 118732281 Ki > 20000 nM T86679 CK24DH 118732282 Ki > 20000 nM T86679 CP78KH 118732283 Ki > 10000 nM T86679 CEO92J 118732284 Ki > 15000 nM T86679 CJ6YF9 118732285 Ki = 60000 nM T86679 CW62JS 118732286 Ki > 20000 nM T86679 CXW9U6 118732287 Ki > 20000 nM T86679 C06FRT 118732288 Ki > 20000 nM T86679 CR2CO8 118732289 Ki > 20000 nM T86679 C94GHE 118732290 Ki > 10000 nM T86679 COJ86X 118732291 Ki > 20000 nM T86679 C1KDT4 118732292 Ki > 20000 nM T86679 C7BO1N 118732293 Ki > 20000 nM T86679 C4EFY5 118732294 Ki > 20000 nM T86679 CKV50L 118732295 Ki > 10000 nM T86679 CT3Q9E 118732296 Ki > 20000 nM T86679 CLRK73 118732297 Ki > 20000 nM T86679 CE85HO 118732298 Ki > 20000 nM T86679 C9Y6EK 118732299 Ki > 20000 nM T86679 CNJ1H0 118732300 Ki > 20000 nM T86679 CX6IN3 118732301 Ki > 20000 nM T86679 C4N6ZT 118732302 Ki > 20000 nM T86679 CDAZ14 118732303 Ki > 20000 nM T86679 CZ7TM6 118732304 Ki > 20000 nM T86679 CXZW46 118732305 Ki > 20000 nM T86679 CWX3P4 118732306 Ki > 20000 nM T86679 CXRT76 118732307 Ki > 10000 nM T86679 CK0NS3 118732308 Ki > 20000 nM T86679 CRFJ71 118732309 Ki > 10000 nM T86679 CT90VA 118732971 EC50 = 347 nM T86679 CXM53U 118732972 EC50 = 1480 nM T86679 CF4G3P 118732973 EC50 = 3510 nM T86679 C3E2BJ 118732974 EC50 = 222 nM T86679 C1U2FS 118732975 EC50 = 677 nM T86679 C4YS5J 118732976 EC50 = 1010 nM T86679 CZ7QU0 118732977 EC50 > 30000 nM T86679 CHP93T 118732978 EC50 = 1340 nM T86679 CBT95M 118732979 EC50 = 3150 nM T86679 CZ3X0P 118732980 EC50 = 530 nM T86679 CMDH59 118732981 EC50 = 1110 nM T86679 C7MZ9V 118732982 EC50 = 834 nM T86679 CVS8R0 118734340 EC50 > 10000 nM T86679 C91DBT 118734341 EC50 > 10000 nM T86679 CV1JE8 118734342 EC50 > 10000 nM T86679 C8AB7F 118734343 EC50 > 10000 nM T86679 CLWV70 118734344 EC50 > 10000 nM T86679 CP7SE9 118734345 EC50 = 9287 nM T86679 CC0RE9 118734346 EC50 = 9352 nM T86679 CV6X3F 118734347 EC50 = 7130 nM T86679 CN8RI9 118734348 EC50 > 10000 nM T86679 CEZ86B 118734349 EC50 > 10000 nM T86679 C1QPJ3 118734350 EC50 > 10000 nM T86679 CFH92R 118734351 EC50 > 10000 nM T86679 CR8FT9 118734352 EC50 > 10000 nM T86679 C8Y7QW 118734353 EC50 > 10000 nM T86679 CR3Y1J 118734354 EC50 > 10000 nM T86679 C5DL3X 118734355 EC50 > 10000 nM T86679 CYB49C 118734356 EC50 > 10000 nM T86679 CZE09N 118734357 EC50 > 10000 nM T86679 CB7J1G 118734358 EC50 > 10000 nM T86679 C79RHZ 118734359 EC50 > 10000 nM T86679 CSAH95 118734360 EC50 > 10000 nM T86679 C1CBG3 118734361 EC50 > 10000 nM T86679 CN9S1Y 118734362 EC50 > 10000 nM T86679 C5SQA1 118734363 EC50 > 10000 nM T86679 CDVO89 118734364 EC50 > 10000 nM T86679 CQ73IF 118734365 EC50 > 10000 nM T86679 C43VAO 118734366 EC50 > 10000 nM T86679 C4NQV6 118734367 EC50 > 10000 nM T86679 CGF84C 118734368 EC50 > 10000 nM T86679 C94UXF 118734369 EC50 > 10000 nM T86679 CU0K8H 118734370 EC50 > 10000 nM T86679 CPY5O0 118734371 EC50 > 10000 nM T86679 CLI1V7 118734372 EC50 = 927 nM T86679 CX08QC 118734373 EC50 > 10000 nM T86679 CD3BV5 118734374 EC50 = 866 nM T86679 C58VBC 118734375 EC50 > 10000 nM T86679 C0U1NA 118734376 EC50 = 389 nM T86679 CZH87J 118734377 EC50 > 10000 nM T86679 C0DK6X 122574669 IC50 = 640 nM T86679 C5UO7Q 122574772 IC50 = 150 nM T86679 C9OR6D 127025959 EC50 = 125892.54 nM T86679 CXG31M 127026188 Ki = 1470 nM T86679 C0MWD8 127026257 EC50 = 331131.12 nM T86679 C5EW3U 127030064 Ki = 847.3 nM T86679 C6WNP3 127030364 Ki = 29.34 nM T86679 C1Q0SH 127030660 Ki = 728.1 nM T86679 CW52ET 127031266 Ki = 11.4 nM T86679 CK0L8R 127033039 Ki = 20.6 nM T86679 CH57JY 127033325 Ki = 29.71 nM T86679 CQN50M 127033645 Ki = 0.5 nM T86679 C16QEM 127034213 Ki = 108 nM T86679 CJ8K1T 127034214 Ki = 85.6 nM T86679 C2VWT7 127034216 Ki = 276.9 nM T86679 C2BM4D 127035624 IC50 > 30000 nM T86679 CFJ95C 127035625 IC50 > 30000 nM T86679 CPY0S3 127035626 IC50 = 4360 nM T86679 CDWC03 127035803 IC50 > 30000 nM T86679 CH41BT 127035804 IC50 > 30000 nM T86679 C7AHR2 127035805 IC50 > 30000 nM T86679 C92RXW 127035806 IC50 = 7617 nM T86679 CGD59Y 127035832 IC50 > 30000 nM T86679 CX29PN 127035833 IC50 > 30000 nM T86679 C4Y3XI 127035834 IC50 > 30000 nM T86679 CJM9Z1 127036437 IC50 > 30000 nM T86679 CM63GQ 127036438 IC50 > 30000 nM T86679 C59HYJ 127036640 IC50 > 30000 nM T86679 CJ52XA 127036641 IC50 > 30000 nM T86679 CX9H5M 127036642 IC50 > 30000 nM T86679 C4F2WP 127036740 IC50 > 30000 nM T86679 C3QVM7 127036741 IC50 > 30000 nM T86679 C3E7ZT 127036742 IC50 > 30000 nM T86679 CGM30I 127036810 IC50 > 30000 nM T86679 CR7OT4 127036811 IC50 > 30000 nM T86679 CR58OX 127036812 IC50 > 30000 nM T86679 C65YKX 127036844 IC50 = 11800 nM T86679 CLCF05 127036845 IC50 > 30000 nM T86679 C5K3MR 127036846 IC50 > 30000 nM T86679 CB8HG0 127036933 IC50 > 30000 nM T86679 C1MS0C 127036976 IC50 > 30000 nM T86679 CQR43P 127036977 IC50 > 30000 nM T86679 C2YT3C 127038355 Ki = 3190 nM T86679 C3CMX4 127038356 Ki = 1740 nM T86679 CB5F1H 127038752 Ki = 680 nM T86679 CR3A5Y 127038753 Ki = 2191 nM T86679 CUD27T 127040064 Ki = 8240 nM T86679 CY4G8A 127040403 Ki > 30000 nM T86679 C9OG1N 127040410 Ki = 7490 nM T86679 C8D4GN 127042408 Ki > 30000 nM T86679 CA1XD7 127042409 Ki = 4610 nM T86679 C7ZOD5 127042993 Ki = 1760 nM T86679 C10OFL 127042994 Ki = 9280 nM T86679 CGE9O0 127042995 Ki > 30000 nM T86679 CCV4W8 127042996 Ki = 1760 nM T86679 C4JR2S 127042997 Ki = 1870 nM T86679 C04FIN 127043159 Ki > 1000 nM T86679 CXK89P 127043160 Ki > 1000 nM T86679 CB9Q2K 127043161 Ki > 1000 nM T86679 CD23GH 127043299 Ki > 10000 nM T86679 CAK8N9 127043339 Ki > 1000 nM T86679 C5PBH0 127043340 Ki > 1000 nM T86679 CG8F3I 127043648 Ki > 10000 nM T86679 C93XPB 127043661 Ki > 1000 nM T86679 CZ5BA7 127043662 Ki > 500 nM T86679 C63QSD 127043663 Ki = 663 nM T86679 CKG3S7 127043664 Ki = 338 nM T86679 C57BHD 127043668 Ki = 853 nM T86679 C9JY6M 127043669 Ki = 131 nM T86679 CH8S0Y 127043671 Ki > 1000 nM T86679 CU6I9L 127043672 Ki > 1000 nM T86679 CQVE62 127043673 Ki > 1000 nM T86679 C1J3PR 127043818 Ki > 10000 nM T86679 C8V5EN 127043828 Ki = 109 nM T86679 C1PXL8 127043829 Ki = 337 nM T86679 CN46BI 127043830 Ki > 1000 nM T86679 COW15S 127043831 Ki > 1000 nM T86679 C2HWP1 127043995 Ki > 1000 nM T86679 CMJL86 127044142 Ki > 10000 nM T86679 CYS6Z4 127044283 Ki > 10000 nM T86679 CC6MG4 127044514 Ki > 10000 nM T86679 CW18JP 127044515 Ki > 10000 nM T86679 C4O7WX 127044516 Ki > 10000 nM T86679 C3KQS4 127044517 Ki > 10000 nM T86679 CE1A4H 127044518 Ki > 10000 nM T86679 CQJ71U 127044681 Ki > 10000 nM T86679 CS0M2P 127044784 Ki > 1000 nM T86679 C7V4HX 127044785 Ki > 10000 nM T86679 CLXU52 127044795 Ki > 10000 nM T86679 C5FC3T 127044855 Ki > 10000 nM T86679 CB35MD 127045017 Ki > 1000 nM T86679 CO9LP5 127045018 Ki > 1000 nM T86679 C87ISU 127045019 Ki > 1000 nM T86679 C8W3FJ 127045020 Ki > 1000 nM T86679 CK0ST8 127045021 Ki > 1000 nM T86679 C53KHG 127045164 Ki > 10000 nM T86679 C5LC0U 127045165 Ki > 10000 nM T86679 CGS9B5 127045166 Ki > 10000 nM T86679 C8NV5Y 127045167 Ki > 1000 nM T86679 C2R9PY 127045168 Ki > 1000 nM T86679 C0RMT7 127045169 Ki > 1000 nM T86679 C7I3NV 127045170 Ki > 1000 nM T86679 CRF57W 127045471 Ki > 1000 nM T86679 CW6B7M 127045472 Ki > 1000 nM T86679 C7FH4S 127045473 Ki > 1000 nM T86679 C9QIC7 127045630 Ki > 1000 nM T86679 C6UK3Q 127045631 Ki > 1000 nM T86679 CQL9K1 127045632 Ki > 1000 nM T86679 C8MT9L 127045699 IC50 = 354 nM T86679 C02HYP 127045700 IC50 = 421 nM T86679 C6VU1I 127045701 IC50 = 152 nM T86679 C4MQU2 127045909 IC50 = 395 nM T86679 CQ1IB0 127045910 IC50 = 633 nM T86679 CDHL50 127046050 IC50 = 293 nM T86679 CH8W3C 127046493 IC50 = 512 nM T86679 COE1R5 127046494 IC50 = 112 nM T86679 CNH42R 127051230 Ki > 30000 nM T86679 C97UBL 127051231 Ki > 30000 nM T86679 CZ9NH5 127051849 Ki > 30000 nM T86679 C4A3IX 127051850 Ki > 30000 nM T86679 C8ACT1 127051851 Ki > 30000 nM T86679 CY2B7M 127051852 Ki > 30000 nM T86679 CPN29G 127052152 Ki > 30000 nM T86679 CB6R7Z 127052168 Ki > 30000 nM T86679 C1TJ7B 132578491 Ki > 1000 nM T86679 C5CKG0 132578492 Ki > 300 nM T86679 CVS8H1 132578493 Ki > 1000 nM T86679 CKIA45 132933622 IC50 > 30000 nM T86679 C02UQE 132941757 Ki = 500 nM T86679 CJ54MF 132991405 IC50 = 313 nM T86679 C75XIA 132991406 IC50 = 452 nM T86679 C3UC1T 134132667 IC50 = 47 nM T86679 C2I7AE 134132684 IC50 = 482 nM T86679 CHSK61 134133787 IC50 = 95 nM T86679 CR38DS 134138275 IC50 = 24 nM T86679 C7WPX1 134138322 IC50 = 553 nM T86679 CV38YZ 134138961 IC50 = 283 nM T86679 CIAY28 134139825 IC50 = 632 nM T86679 C2KSZ9 134142435 IC50 = 103 nM T86679 C5ZAD2 134142611 IC50 = 25 nM T86679 CR1YQ6 134142843 Ki > 30000 nM T86679 C3L2PZ 134147788 IC50 = 32 nM T86679 CRA5O4 134147994 IC50 = 1768 nM T86679 C4MDF2 134148336 IC50 = 1000 nM T86679 CPI01N 134149255 IC50 = 389 nM T86679 CNET28 134151346 IC50 = 323 nM T86679 C1JK6T 134152846 IC50 = 18 nM T86679 C20RNA 134157761 IC50 = 185 nM T86679 C08ZQW 135404340 Ki = 1900 nM T86679 C9WD5K 135405767 IC50 > 1000 nM T86679 C2ATW9 135409793 Ki = 6660 nM T86679 C5T2ZE 135409960 IC50 > 1000 nM T86679 C8ZY2A 135414399 Ki = 3700 nM T86679 C6G0HA 135416050 Ki = 78 nM T86679 CI0HT3 135416055 Ki = 130 nM T86679 C1IEY0 135418256 IC50 = 2700 nM T86679 C0C5IU 135418454 Ki = 6 nM T86679 C0Z8RU 135421343 Ki > 1000 nM T86679 CW16MF 135421366 Ki = 74 nM T86679 CUA67Z 135423046 Ki = 350 nM T86679 CD1SB0 135424850 Ki = 1100 nM T86679 CT85YL 135428628 Ki = 2200 nM T86679 CY9QI4 135428630 Ki = 2000 nM T86679 C7P2ME 135428645 Ki = 580 nM T86679 C5OZ0L 135428653 Ki = 3100 nM T86679 CI4Z3R 135430228 Ki = 85 nM T86679 CZA5F9 135436760 Ki > 1000 nM T86679 C6HN3Z 135438480 Ki = 17800 nM T86679 CI4S7C 135440168 Ki = 41 nM T86679 CR9W5J 135440414 Ki > 1000 nM T86679 C1UNH9 135440428 Ki = 185 nM T86679 C5YUC2 135443302 Ki = 235 nM T86679 CO87CV 135443324 Ki = 569 nM T86679 CWD8M7 135443353 Ki = 39 nM T86679 C4KLO0 135443378 Ki = 13 nM T86679 CG9IK2 135444614 Ki = 21 nM T86679 C9UCG0 135448286 Ki = 86 nM T86679 C0B1XV 135454766 IC50 > 1000 nM T86679 C4DUN5 135464144 Ki = 1030 nM T86679 CU14JT 135465774 Ki = 50 nM T86679 C1F5CA 135465776 Ki = 70 nM T86679 C04XNV 135465778 Ki = 90 nM T86679 CBV8I2 135465784 Ki = 342 nM T86679 C7E2CQ 135465796 Ki = 132 nM T86679 C0YZ3B 135470411 Ki > 1000 nM T86679 CPQ3J6 135477916 IC50 > 1000 nM T86679 CK52RH 135483531 Ki = 93 nM T86679 CTU21N 135483619 IC50 > 1000 nM T86679 CJ91TZ 135484407 IC50 > 10000 nM T86679 CI8R0L 135485985 Ki = 51 nM T86679 CE26MK 135486084 Ki = 2065 nM T86679 CH0AR8 135486118 Ki = 303 nM T86679 CF13KU 135489505 Ki = 2100 nM T86679 CVG5M0 135493238 Ki = 58 nM T86679 CCX3D7 135493268 Ki = 35 nM T86679 CF06CK 135493272 Ki = 103 nM T86679 CS3OC8 135493279 Ki = 12 nM T86679 C9RS5H 135493280 Ki = 160 nM T86679 CEI8W7 135493281 Ki = 28 nM T86679 C25QGD 135493285 Ki = 1628 nM T86679 CN10IO 135493286 Ki = 59 nM T86679 C7O1NS 135493290 Ki > 1000 nM T86679 CV4X0H 135493292 Ki = 51 nM T86679 C5OK7A 135499926 Ki = 90 nM T86679 CU8W5N 135508372 IC50 > 1000 nM T86679 CTB6R7 135515408 IC50 = 9400 nM T86679 CFQ38U 135515507 Ki = 70 nM T86679 C46YPU 135519330 IC50 > 1000 nM T86679 CG64XS 135522362 Ki = 76 nM T86679 C1E2ZK 135522363 Ki = 96 nM T86679 C2CL8J 135522364 Ki = 81 nM T86679 C2AHQ6 135522367 Ki = 18 nM T86679 CF9XI7 135522375 Ki = 12 nM T86679 C4NG7Y 135522388 Ki = 20 nM T86679 C9A7QL 135522390 Ki = 86 nM T86679 CUNG36 135522391 Ki = 55 nM T86679 CFJ8P2 135525108 IC50 > 10000 nM T86679 CQ9ZO5 135528632 Ki = 4.9 nM T86679 C2WJI6 135529341 Ki > 1000 nM T86679 C7ARF8 135529362 Ki > 1000 nM T86679 C2V3CX 135529371 Ki = 100 nM T86679 CVXF23 135529372 Ki = 53 nM T86679 CJ86ZY 135529373 Ki = 78 nM T86679 CESZ83 135529396 Ki = 66 nM T86679 CJ4Y1H 135529398 Ki = 111 nM T86679 C51PIY 135543600 Ki = 838 nM T86679 CF3UQ4 135543624 EC50 = 12 nM T86679 C6WLJ3 135544018 IC50 > 10000 nM T86679 C1K5QE 135544028 IC50 > 10000 nM T86679 CR6X3F 135544059 IC50 > 10000 nM T86679 C38LZC 135545353 IC50 > 1000 nM T86679 C5Y9WX 135546648 Ki = 88 nM T86679 CESD69 135546649 Ki = 19 nM T86679 CUI90X 135546657 Ki = 38 nM T86679 C5KX8N 135546658 Ki = 207 nM T86679 C9OCX4 135610070 Ki = 18 nM T86679 C8LBZ5 135624236 IC50 > 10000 nM T86679 C3VK1O 135633267 Ki = 602.4 nM T86679 CJO5S1 135633268 Ki = 350.5 nM T86679 C7KW6I 135678052 Ki = 7 nM T86679 C6GI3C 135738646 IC50 < 100 nM T86679 C67BTG 135738649 IC50 > 1500 nM T86679 CD6GS7 135738659 IC50 > 2600 nM T86679 CR12ZF 135805568 Ki = 55.6 nM T86679 C62PTQ 135874413 Ki = 15 nM T86679 C87ZQJ 135874414 Ki = 28 nM T86679 C9X1UL 135874415 Ki = 35 nM T86679 CT40VW 135874416 Ki = 14 nM T86679 C1V9TY 135874420 Ki = 12 nM T86679 C1T4GB 135874421 Ki = 48 nM T86679 CFSX68 135874422 Ki = 60 nM T86679 CNLH54 135874423 Ki > 1000 nM T86679 C2FK6J 135874424 Ki = 20 nM T86679 C04YTD 135874425 Ki > 1000 nM T86679 CIQ04D 135874427 Ki > 1000 nM T86679 C6TO4A 135874428 Ki = 65 nM T86679 CO0C5V 135874429 Ki = 28 nM T86679 C9JQ2C 135874430 Ki = 40 nM T86679 CSOV01 135874431 Ki = 56 nM T86679 C75TGS 135874432 Ki = 222 nM T86679 C93GBH 135874433 Ki = 250 nM T86679 CV7US0 135874434 Ki > 1000 nM T86679 CF0SZ2 135915276 Ki = 15 nM T86679 COT8D1 135915277 Ki = 55 nM T86679 C20IDY 135915282 Ki > 600 nM T86679 CB02RD 135915284 Ki > 600 nM T86679 CIVD34 135949027 Ki = 370 nM T86679 C7R9LG 136002185 Ki = 1012 nM T86679 C3BV1J 136002186 Ki = 34 nM T86679 CSBL59 136002187 Ki = 175 nM T86679 CGS18F 136002248 Ki = 9.4 nM T86679 CO62QD 136015813 EC50 = 23.44 nM T86679 CUK9J5 136019511 IC50 > 5000 nM T86679 CBZ1I4 136025838 IC50 > 5000 nM T86679 CCS5F0 136025881 IC50 > 5000 nM T86679 C2VZR6 136025990 IC50 > 5000 nM T86679 CA17MI 136026025 IC50 > 5000 nM T86679 C9SR2V 136026026 IC50 > 5000 nM T86679 C6KNF2 136026027 IC50 > 5000 nM T86679 CO90BT 136026133 IC50 > 5000 nM T86679 CM3YH2 136026181 IC50 > 5000 nM T86679 C38LUX 136036809 Ki > 1000 nM T86679 CQ49LB 136042243 IC50 > 100000 nM T86679 CEHF18 136042327 Ki = 20 nM T86679 C4U7ZM 136042328 Ki = 14.8 nM T86679 CSR0Z3 136042329 Ki = 12 nM T86679 C9C2SF 136042330 Ki = 88 nM T86679 C75CXE 136042331 Ki = 14.1 nM T86679 CS49WL 136042332 Ki = 25 nM T86679 CQ2ZA9 136042333 Ki = 19 nM T86679 CON2J4 136042334 Ki = 22 nM T86679 C5VY2Z 136042335 Ki = 48.98 nM T86679 CTEB06 136042336 Ki > 1000 nM T86679 CJW64L 136042337 Ki = 61 nM T86679 C05QUF 136042338 Ki = 23 nM T86679 C0SX1K 136042339 Ki = 3.5 nM T86679 CQ37GX 136042340 Ki = 4.1 nM T86679 CF3BR5 136042341 Ki = 10 nM T86679 C75XRI 136042342 Ki = 35 nM T86679 CS7HM2 136042343 Ki = 5.5 nM T86679 C3S1WY 136042344 Ki = 22 nM T86679 CR5H4M 136042345 Ki = 76 nM T86679 C29YZE 136042346 Ki = 11.4 nM T86679 CAP1C6 136042347 Ki = 13.4 nM T86679 C5EX7D 136042348 Ki = 87 nM T86679 C4L7GE 136042349 Ki = 30 nM T86679 C9JM7Y 136042350 Ki = 5 nM T86679 CO15GM 136042351 Ki = 14.2 nM T86679 COEZ25 136042352 Ki = 15.9 nM T86679 CGX6H7 136042353 Ki = 8.1 nM T86679 C1W9XD 136042354 Ki = 10.2 nM T86679 CA6TI2 136042355 Ki = 18 nM T86679 CZNC93 136044105 Ki = 46.5 nM T86679 C2A9NB 136044106 Ki = 20.7 nM T86679 C61CMJ 136044107 Ki = 138 nM T86679 CQXL71 136044108 Ki = 125 nM T86679 CF71HS 136044130 Ki = 188 nM T86679 CJ75XH 136068601 IC50 > 5000 nM T86679 CL5B7U 136068602 IC50 > 5000 nM T86679 CU6C4Z 136068688 IC50 > 5000 nM T86679 CSJE87 136068689 IC50 > 5000 nM T86679 C7SLK3 136068716 IC50 > 5000 nM T86679 CZWP52 136068717 IC50 > 5000 nM T86679 CDX2Q0 136068718 IC50 > 5000 nM T86679 CY1RT3 136068719 IC50 > 5000 nM T86679 CU8C3J 136086750 Ki = 1584.89 nM T86679 CI1PK7 136086896 IC50 > 5000 nM T86679 C5HL7K 136086897 IC50 > 5000 nM T86679 C6VLR1 136086898 IC50 > 5000 nM T86679 CL2E0U 136086899 IC50 > 5000 nM T86679 C01GMB 136086900 IC50 > 5000 nM T86679 CA3X5T 136086901 IC50 > 5000 nM T86679 CW49CH 136086902 IC50 > 5000 nM T86679 C4F5WR 136086903 IC50 > 5000 nM T86679 CS58QU 136086904 IC50 > 5000 nM T86679 C4B1TU 136086905 IC50 > 5000 nM T86679 CMOR91 136086906 IC50 > 5000 nM T86679 C3HY9O 136086907 IC50 > 5000 nM T86679 CWF2L1 136086908 IC50 > 5000 nM T86679 CQHW89 136184487 Ki > 1000 nM T86679 C1OU7W 136184488 Ki > 1000 nM T86679 CW2D5Y 136184489 Ki > 1000 nM T86679 CI2YG5 136184490 Ki > 1000 nM T86679 CN6RY1 136184491 Ki > 1000 nM T86679 C8OWD1 136184493 Ki > 1000 nM T86679 CRC2O9 136184494 Ki > 1000 nM T86679 C5EPJ2 136199393 Ki = 31 nM T86679 CF51IY 136228031 Ki > 10000 nM T86679 C5IX2C 136236319 Ki > 10000 nM T86679 CU6MT1 136383804 Ki = 69 nM T86679 CNV4Q9 136396061 Ki = 210 nM T86679 CBDP73 136414898 Ki = 90 nM T86679 CWL69G 136414902 Ki = 12.8 nM T86679 C8K0NO 137175186 Ki = 699.2 nM T86679 CB3NC8 137175187 Ki = 816.7 nM T86679 C9QS4J 137631671 Ki = 650 nM T86679 CSM29H 137632333 Ki = 10000 nM T86679 CQ36UP 137632356 IC50 > 30000 nM T86679 CH5F6G 137632488 EC50 > 60000 nM T86679 C92FIL 137632746 IC50 > 30000 nM T86679 CFWO04 137632925 IC50 > 30000 nM T86679 CJ67UL 137633007 IC50 > 30000 nM T86679 CZ2HV1 137633654 EC50 > 30000 nM T86679 CZC9A2 137633810 IC50 > 30000 nM T86679 C8K7EM 137634052 EC50 = 97.72 nM T86679 C9YB3R 137634085 Ki = 5000 nM T86679 C71MVS 137634444 EC50 = 63.1 nM T86679 C61PXN 137634776 Ki = 24.3 nM T86679 CRGN40 137635666 IC50 > 30000 nM T86679 CYL3X8 137636099 EC50 = 1650 nM T86679 C8H9DB 137636200 Ki = 200 nM T86679 CC9P6O 137636304 Ki = 500 nM T86679 C01OZS 137636323 IC50 > 30000 nM T86679 CS1EO0 137636334 IC50 > 30000 nM T86679 CU9G8K 137636427 IC50 > 30000 nM T86679 C5P9LI 137637451 EC50 > 60000 nM T86679 C53RQW 137637667 IC50 > 30000 nM T86679 C6Q9JG 137637685 Ki = 579 nM T86679 CCTH80 137638080 EC50 = 592 nM T86679 CW4S1V 137638211 IC50 > 30000 nM T86679 CQ8ZL2 137638623 IC50 > 30000 nM T86679 CBM92H 137638964 Ki = 15.1 nM T86679 CZ9QX0 137639459 IC50 > 30000 nM T86679 CTQ67J 137639588 EC50 = 288.4 nM T86679 CMGI82 137639632 Ki = 330 nM T86679 C0SC7L 137640093 IC50 > 30000 nM T86679 CV51BA 137640112 Ki = 7.8 nM T86679 C56BND 137640212 Ki = 102 nM T86679 C45FXO 137641603 EC50 > 30000 nM T86679 CG0DI3 137641858 EC50 = 91.2 nM T86679 C52XDH 137641906 IC50 > 30000 nM T86679 CFW9R5 137641990 EC50 = 2570 nM T86679 CV81KH 137642036 EC50 = 637 nM T86679 CE4C5Y 137642150 IC50 > 30000 nM T86679 CO94EX 137642153 EC50 = 527 nM T86679 CI34WT 137642862 Ki = 23 nM T86679 C7K9ZB 137642980 IC50 > 30000 nM T86679 C76XKJ 137643150 IC50 > 30000 nM T86679 CJQD73 137643164 EC50 = 17.78 nM T86679 CG46DW 137644190 IC50 > 30000 nM T86679 CPR72G 137644224 IC50 > 30000 nM T86679 C4R0OC 137644481 IC50 > 30000 nM T86679 CI7B3F 137645065 EC50 > 60000 nM T86679 CGLI82 137645223 EC50 > 60000 nM T86679 CF09IY 137645275 IC50 > 30000 nM T86679 CCL76A 137645670 Ki = 79 nM T86679 CDBT79 137645728 IC50 > 30000 nM T86679 C95UJV 137645798 IC50 > 30000 nM T86679 CJ20CU 137645935 Ki = 1400 nM T86679 C8YN3Q 137646655 EC50 = 446.68 nM T86679 CER23T 137646828 EC50 = 75.86 nM T86679 CGL83H 137647102 IC50 > 30000 nM T86679 CY2H5K 137647216 Ki = 120 nM T86679 CC0UF1 137647420 EC50 = 408 nM T86679 CT91AP 137648111 IC50 > 30000 nM T86679 CCA7I4 137648143 IC50 > 30000 nM T86679 C1AIP8 137648928 EC50 = 235 nM T86679 CS3DT1 137649083 EC50 = 18.62 nM T86679 C62KVF 137649307 Ki = 96.2 nM T86679 C5CJI7 137649458 Ki = 100 nM T86679 CWH89G 137649841 EC50 = 158.49 nM T86679 CIE03Y 137650221 EC50 = 2140 nM T86679 CN5QM6 137650340 Ki = 461 nM T86679 CSO92A 137650430 Ki = 51 nM T86679 C9W3PX 137650461 EC50 = 616.6 nM T86679 CIM50G 137650899 EC50 = 1930 nM T86679 CXCA79 137650918 EC50 = 223.87 nM T86679 C26YKP 137651319 IC50 > 30000 nM T86679 CEAU34 137651531 EC50 > 30000 nM T86679 C13AMI 137651532 IC50 > 30000 nM T86679 C9M7QE 137651747 EC50 = 2230 nM T86679 C6Z1HJ 137651756 EC50 = 12800 nM T86679 CVS93H 137652383 EC50 > 60000 nM T86679 C8T2HN 137652475 EC50 = 467.74 nM T86679 C79MDG 137652737 Ki = 349.1 nM T86679 CJ24ZP 137653290 IC50 > 30000 nM T86679 CHYT41 137653409 EC50 = 60.26 nM T86679 CJ1R9K 137653588 EC50 > 30000 nM T86679 CA24YS 137656139 EC50 > 60000 nM T86679 CX21IZ 137656644 Ki = 647 nM T86679 C28GAV 137656845 EC50 = 147.91 nM T86679 CJUE21 137656913 EC50 = 20000 nM T86679 C08KJH 137657382 EC50 > 60000 nM T86679 CH8PL9 137657570 EC50 > 60000 nM T86679 CNTX97 137657841 EC50 = 1290 nM T86679 CJ8BC7 137657926 EC50 = 1961 nM T86679 CQ9BR1 137658051 IC50 > 30000 nM T86679 CBC31H 137658387 IC50 > 30000 nM T86679 CU40KY 137658586 Ki = 59.4 nM T86679 CH9A8M 137658761 EC50 = 3740 nM T86679 CV7UE3 137659204 IC50 > 30000 nM T86679 CY67UM 137659236 IC50 > 30000 nM T86679 C7VNS4 137659441 EC50 = 1100 nM T86679 CT23EA 137659930 IC50 > 30000 nM T86679 C1NZL8 137659963 IC50 > 30000 nM T86679 CIDG46 137660466 Ki = 51.2 nM T86679 CQW9O4 137660519 Ki = 140 nM T86679 C3Y2IZ 137661132 EC50 = 2390 nM T86679 CFUM75 137661322 EC50 > 60000 nM T86679 C26LVX 137661505 EC50 = 35.48 nM T86679 C1DL4J 137661670 EC50 > 30000 nM T86679 COM9G6 137661811 IC50 > 30000 nM T86679 CD1Z9C 137661874 Ki = 23 nM T86679 CT26DO 137662145 IC50 > 30000 nM T86679 CP02WU 139030524 EC50 > 1000 nM T86679 CU3PW1 139248507 Ki > 1000 nM T86679 CT1H6B 139248508 Ki > 1000 nM T86679 CUIN96 139248509 Ki > 1000 nM T86679 CW74BD 141536950 IC50 > 30000 nM T86679 CV48QA 142752615 IC50 > 10000 nM T86679 CBV2L5 145436760 IC50 = 75 nM T86679 CK15TH 145436761 IC50 = 13.2 nM T86679 C6KOB8 145436762 IC50 = 14 nM T86679 CM7J2Q 145436763 IC50 = 4.21 nM T86679 CSQL37 145436764 IC50 = 8.96 nM T86679 CNP52A 145436765 IC50 = 112 nM T86679 C6OFP7 145436766 IC50 = 95 nM T86679 CSQ8U5 145436767 IC50 = 109 nM T86679 C4PZ5S 145436769 IC50 = 82 nM T86679 CI75YJ 145949481 IC50 = 91 nM T86679 CLMF57 145952391 Ki = 1.82 nM T86679 C2GVM4 145954098 IC50 = 547 nM T86679 CQ9G0K 145954398 IC50 = 389 nM T86679 C3RU6S 145954471 IC50 = 120 nM T86679 CZX79R 145954995 Ki > 30000 nM T86679 CHYQ29 145958145 Ki = 1.047 nM T86679 CC0OX1 145958464 IC50 = 4571 nM T86679 CH7G6S 145960536 IC50 = 1810 nM T86679 C9PT5Q 145960667 IC50 = 1105 nM T86679 C3BY8E 145960746 IC50 = 5013 nM T86679 CWSM81 145960813 IC50 = 72 nM T86679 C5D6AI 145960873 IC50 = 4380 nM T86679 C62JCL 145960933 Ki = 230 nM T86679 CRBY29 145961339 IC50 = 3725 nM T86679 C02OQR 145961748 IC50 = 4017 nM T86679 C1O0GQ 145961937 IC50 = 784 nM T86679 CCB0Y2 145961997 IC50 = 3516 nM T86679 CT8UO0 145962202 IC50 = 2387 nM T86679 C3M7ZN 145962234 IC50 > 10000 nM T86679 CVA89T 145962310 IC50 = 7524 nM T86679 CD6X5O 145962355 IC50 = 2622 nM T86679 C86APL 145962364 IC50 = 2072 nM T86679 CH5DS7 145962529 IC50 = 134 nM T86679 C4NXC1 145962657 IC50 > 10000 nM T86679 C9UYI6 145963230 IC50 = 358 nM T86679 C5MD4S 145963661 IC50 = 5538 nM T86679 C9E0UX 145964230 Ki = 27.9 nM T86679 CS0O1Z 145964662 Ki = 7 nM T86679 C86XTA 145965011 EC50 = 347 nM T86679 C01PVB 145965471 EC50 = 11.7 nM T86679 CYZ05R 145967103 EC50 = 332 nM T86679 C1ER6I 145967791 Ki = 5.9 nM T86679 CLD46J 145968949 EC50 = 182 nM T86679 CY20LR 145970075 Ki = 3.3 nM T86679 CYX65N 145971695 Ki = 1.318 nM T86679 CP10LJ 145971798 Ki = 11.6 nM T86679 C8J7FL 145971923 IC50 = 33 nM T86679 CNU0Q9 145972065 EC50 = 51 nM T86679 CZJA45 145972655 IC50 = 2773 nM T86679 CE23KG 145973077 EC50 = 9.5 nM T86679 CV9OM2 145973260 Ki = 5000 nM T86679 CBT7E9 145973326 Ki = 7.82 nM T86679 CJH7D0 145974358 EC50 = 12.7 nM T86679 CB96ZI 145975418 Ki = 24.4 nM T86679 CKMZ02 145975919 EC50 = 38 nM T86679 C9TLO2 145976032 EC50 = 84 nM T86679 CZI4H3 145976828 Ki = 7.45 nM T86679 CI2HN1 145977111 Ki = 1.83 nM T86679 CM1R0J 145977114 EC50 = 211 nM T86679 CBO9F4 145977469 EC50 = 139 nM T86679 CA1YE3 145979018 Ki = 298 nM T86679 C9VTO3 145979285 Ki = 275 nM T86679 C8DW3E 145979590 Ki > 1000 nM T86679 C5SZN2 145979632 Ki > 10000 nM T86679 C9T3DG 145980225 Ki > 1000 nM T86679 COK2V5 145980546 Ki > 10000 nM T86679 CO3Y8B 145980553 Ki > 10000 nM T86679 CP92RY 145980571 Ki > 10000 nM T86679 CBCH87 145980626 Ki > 1000 nM T86679 C7NJH2 145980712 Ki > 10000 nM T86679 CHU27O 145980918 Ki > 1000 nM T86679 CMFW02 145980971 Ki = 10000 nM T86679 CDM63O 145981315 Ki > 10000 nM T86679 C0T4WK 145981370 Ki = 113 nM T86679 CHQ73C 145981492 Ki > 10000 nM T86679 CA9R1X 145981583 Ki > 10000 nM T86679 CK14YF 145981625 Ki > 1000 nM T86679 CB1Y4K 145981689 Ki = 452 nM T86679 CX02DQ 145981864 Ki > 10000 nM T86679 CNTY13 145982075 Ki = 1000 nM T86679 CAI53J 145982270 Ki > 10000 nM T86679 CHSJ14 145982423 Ki > 30000 nM T86679 C8RT4W 145982945 Ki > 10000 nM T86679 C9CG6I 145984161 Ki > 10000 nM T86679 CUM74P 145984609 Ki > 10000 nM T86679 C9VDN3 145985635 Ki > 10000 nM T86679 CHS8P7 145986422 Ki = 193 nM T86679 C19BNU 145986670 Ki > 10000 nM T86679 CS7D6N 145986838 Ki = 340 nM T86679 C23OKD 145986973 Ki > 1000 nM T86679 CQ9AK0 145987082 Ki > 10000 nM T86679 CJ70FS 145987226 Ki > 3000 nM T86679 C78MWI 145987354 Ki = 126 nM T86679 C05IZF 145987813 Ki > 10000 nM T86679 CGV37C 145987819 Ki = 3720 nM T86679 CYB95S 145987987 Ki > 1000 nM T86679 C0AF1D 145988094 Ki > 10000 nM T86679 CMD74V 145988733 Ki > 10000 nM T86679 CV6CA4 145988962 Ki = 215 nM T86679 CEM2L0 145989440 Ki > 30000 nM T86679 CP3G4S 145989441 Ki > 1000 nM T86679 CVS17Y 145989611 Ki > 10000 nM T86679 CB9GL1 145989764 Ki > 10000 nM T86679 CB6U5A 145989810 Ki = 578 nM T86679 C4I1EY 145990207 Ki > 10000 nM T86679 CZP5T3 145990301 Ki > 10000 nM T86679 CJ0A5L 145990511 Ki > 10000 nM T86679 CHV8C9 145990554 Ki > 3000 nM T86679 C3H2ZP 145990725 Ki > 10000 nM T86679 CJ30YT 145990769 Ki > 10000 nM T86679 C2Y8PA 145990926 Ki > 10000 nM T86679 CV5XO6 145991048 Ki > 10000 nM T86679 C6ZYL7 145991283 Ki = 6060 nM T86679 C9YO2T 145991303 Ki > 10000 nM T86679 CN7A1X 145991427 Ki > 10000 nM T86679 C26OBR 145991489 Ki = 306 nM T86679 CUP48Y 145991545 Ki > 10000 nM T86679 C8QT3X 145991607 Ki > 10000 nM T86679 C7K5ZQ 145991651 Ki > 30000 nM T86679 C8SI9A 145991749 Ki > 3000 nM T86679 C2CB3J 145991827 Ki > 10000 nM T86679 CGH8T9 145992005 Ki > 1000 nM T86679 C3QHT6 145992189 Ki > 10000 nM T86679 CLS8P3 145992357 Ki > 1000 nM T86679 C0NUC8 145992378 Ki > 1000 nM T86679 C1MU4D 145992652 Ki > 10000 nM T86679 CB85AS 145992677 Ki > 10000 nM T86679 C94OJE 145992790 Ki > 10000 nM T86679 C7B3FY 145992928 Ki > 10000 nM T86679 C47DOA 145993092 Ki > 10000 nM T86679 C9KE3Y 145993107 Ki = 66.3 nM T86679 CW7AK5 145993147 Ki = 911 nM T86679 CQ5Y3F 145993331 Ki = 862 nM T86679 CZOR31 145993511 Ki > 10000 nM T86679 CTE42N 145993653 Ki > 1000 nM T86679 CO54SG 145993861 Ki = 179 nM T86679 C6A3RN 145993941 Ki > 10000 nM T86679 C0EY3Q 145994002 Ki > 1000 nM T86679 CO69HC 145994068 Ki > 10000 nM T86679 C72SMW 145994175 Ki > 30000 nM T86679 CE07TR 145994259 Ki = 10000 nM T86679 CJA34O 154701278 Ki = 8.73 nM T86679 C14XVK 155510489 IC50 > 30000 nM T86679 C27RDY 155511376 Ki = 15.14 nM T86679 CD52TC 155511687 IC50 > 30000 nM T86679 CLZD15 155511760 Ki = 49.2 nM T86679 CPMN94 155511844 EC50 > 1000 nM T86679 CM5ZA9 155512438 Ki = 1.28 nM T86679 C3G6WQ 155512463 IC50 = 4700 nM T86679 CX96QM 155512576 Ki > 10000 nM T86679 C4A1VC 155513258 Ki = 588 nM T86679 CGS27D 155513515 IC50 > 30000 nM T86679 CJ81VL 155513866 IC50 > 10000 nM T86679 CUB2C9 155514153 EC50 > 1000 nM T86679 C38LUS 155514209 IC50 > 30000 nM T86679 CKVM85 155514248 Ki > 1000 nM T86679 CR85FY 155514357 Ki > 3000 nM T86679 CQ7GR6 155514463 IC50 > 30000 nM T86679 CRF2B1 155514696 EC50 > 1000 nM T86679 CJP23L 155514761 IC50 = 220 nM T86679 CN8E1J 155514860 Ki = 0.397 nM T86679 CP6C5S 155514957 Ki = 0.403 nM T86679 CEA7B6 155515166 IC50 = 145 nM T86679 CLJ7Y3 155515226 Ki > 10000 nM T86679 CP45UX 155515805 IC50 = 135 nM T86679 CNV02U 155516016 Ki > 1000 nM T86679 CT18NO 155516071 IC50 = 9658 nM T86679 CN36DG 155516146 Ki = 157 nM T86679 CLX4D7 155516277 Ki = 0.432 nM T86679 CO9PI2 155516509 Ki > 1000 nM T86679 C5QJ4R 155516939 Ki > 1000 nM T86679 CO79ET 155517038 IC50 = 3300 nM T86679 CAH53U 155517120 Ki > 1000 nM T86679 CK8FH7 155517501 IC50 > 10000 nM T86679 CR59VH 155517789 IC50 > 30000 nM T86679 CSQL20 155517938 Ki = 643 nM T86679 C0CR9Q 155518147 Ki = 6.08 nM T86679 CI2Q9O 155518555 IC50 = 430 nM T86679 C3SAR7 155519016 Ki > 300 nM T86679 CP74IJ 155519148 IC50 > 30000 nM T86679 C0EAY4 155519375 EC50 > 1000 nM T86679 CX1MO3 155519551 EC50 > 1000 nM T86679 C5NTJ8 155519776 IC50 > 30000 nM T86679 CNLA72 155519860 IC50 = 30 nM T86679 C72OJY 155519986 IC50 > 30000 nM T86679 C8N1CQ 155520115 IC50 > 30000 nM T86679 C8I2DC 155520204 IC50 = 4900 nM T86679 C7AHD8 155520492 IC50 = 42 nM T86679 CZ1S5N 155520662 IC50 > 30000 nM T86679 CY25CV 155520663 Ki > 1000 nM T86679 C7R8UB 155520744 Ki > 1000 nM T86679 CRBE64 155520811 Ki > 1000 nM T86679 CPL4Q7 155520955 IC50 = 17330 nM T86679 CXW82M 155520967 Ki > 300 nM T86679 C6A4UH 155521103 IC50 > 30000 nM T86679 CAC2H5 155521304 Ki > 1000 nM T86679 CS2GJ8 155521355 IC50 > 30000 nM T86679 C4X3KN 155521394 IC50 = 200 nM T86679 C25KBM 155521478 IC50 > 30000 nM T86679 CI9U3X 155521508 IC50 = 180 nM T86679 CYW7Q0 155521543 Ki = 0.137 nM T86679 CXD9G0 155521637 Ki = 1000 nM T86679 CW29KY 155521694 IC50 > 30000 nM T86679 C2V8SU 155521773 Ki > 1000 nM T86679 CW0Z8S 155521875 IC50 = 1600 nM T86679 CHTX98 155522541 Ki = 0.894 nM T86679 C73IUC 155522786 Ki = 61.5 nM T86679 CB79ON 155522797 IC50 = 390 nM T86679 CGJ0W4 155522875 IC50 > 30000 nM T86679 CBW5G4 155522899 IC50 > 30000 nM T86679 CU57IK 155522968 IC50 = 250 nM T86679 CJ3IV5 155523200 IC50 = 200 nM T86679 C71PEJ 155523243 IC50 = 1700 nM T86679 C3SJ9B 155523748 IC50 > 30000 nM T86679 CK8RS0 155523968 Ki = 0.421 nM T86679 C4ZIH2 155524032 Ki = 0.159 nM T86679 C6WO5S 155524137 Ki = 29.6 nM T86679 CD24BF 155524446 Ki > 1000 nM T86679 C8E3HR 155524516 Ki = 48.2 nM T86679 CYSK39 155525038 IC50 > 30000 nM T86679 CZX2N4 155525050 Ki = 0.616 nM T86679 C1WZX5 155525062 Ki > 1000 nM T86679 CN1C6R 155525265 IC50 > 30000 nM T86679 C8QIF6 155525396 Ki = 79.43 nM T86679 C78DHT 155525494 IC50 > 30000 nM T86679 CXP27L 155525648 IC50 = 1300 nM T86679 CR6A7N 155525747 IC50 > 30000 nM T86679 CY0W2Z 155525787 Ki > 1000 nM T86679 CX45HJ 155525800 IC50 > 10000 nM T86679 CPX93A 155526277 IC50 = 39 nM T86679 CHW01V 155526352 IC50 = 200 nM T86679 C6AE2B 155526484 IC50 = 14 nM T86679 C2N8MD 155527056 IC50 = 130 nM T86679 CBAK91 155527112 Ki > 3000 nM T86679 CS9U0T 155527740 IC50 > 30000 nM T86679 C86KIL 155527931 Ki > 1000 nM T86679 C9CIO6 155527939 Ki = 11.24 nM T86679 C3KA0S 155528136 Ki = 0.342 nM T86679 CQHK94 155528396 EC50 > 1000 nM T86679 CR5E7W 155528403 Ki > 1000 nM T86679 C4OL2X 155528461 Ki > 300 nM T86679 CAR75Z 155528717 Ki = 1.91 nM T86679 CZ53GQ 155528757 Ki > 10000 nM T86679 CGX6S4 155529530 Ki > 1000 nM T86679 C19JPC 155529645 IC50 = 50 nM T86679 CZ9YC8 155529872 Ki = 0.215 nM T86679 C7WDL3 155530036 Ki > 1000 nM T86679 CVE30Z 155530257 Ki = 0.629 nM T86679 C34VYA 155530298 Ki > 1000 nM T86679 CQT8O2 155530381 Ki = 0.706 nM T86679 C78JZY 155530514 Ki = 0.148 nM T86679 CY3QH2 155530781 Ki > 1000 nM T86679 CN87UW 155530961 Ki = 20 nM T86679 C2YDZ8 155531112 Ki > 300 nM T86679 C5X1QC 155531135 Ki > 1000 nM T86679 C13NXZ 155531338 Ki > 1000 nM T86679 CNVU03 155531548 IC50 > 30000 nM T86679 C3XQ9S 155531570 IC50 > 30000 nM T86679 C4A3DX 155531727 Ki = 3.22 nM T86679 C16ZTW 155531840 Ki = 6.91 nM T86679 C42MHY 155531922 Ki = 37.42 nM T86679 C0NXR4 155531946 Ki = 575 nM T86679 CQI01K 155531990 Ki = 0.632 nM T86679 C7A9BH 155532173 IC50 > 30000 nM T86679 C21MLU 155532274 Ki = 0.234 nM T86679 CXMC14 155532373 Ki > 1000 nM T86679 CVI21H 155532514 Ki = 1.02 nM T86679 C86SCT 155532773 IC50 > 30000 nM T86679 CQ96YB 155532918 Ki = 10000 nM T86679 C9EU2D 155533104 IC50 > 30000 nM T86679 CBM2O9 155533281 Ki = 521 nM T86679 CY8O6B 155533349 Ki > 3000 nM T86679 CCG1K2 155533519 EC50 > 1000 nM T86679 C8FCH7 155533611 Ki > 1000 nM T86679 CHQ27S 155533818 IC50 = 1700 nM T86679 CY5Q7X 155533829 Ki = 17.03 nM T86679 C7E5OP 155533880 Ki > 10000 nM T86679 C9WO1Z 155533882 Ki > 1000 nM T86679 CH54UR 155534188 Ki > 10000 nM T86679 CKM60Q 155534231 Ki > 1000 nM T86679 CW8FN0 155534473 IC50 > 30000 nM T86679 C9QV4W 155534659 IC50 > 30000 nM T86679 C0R3PA 155534717 Ki > 1000 nM T86679 C4NU8B 155534836 Ki = 0.644 nM T86679 CIH0T5 155535400 Ki > 1000 nM T86679 CRQW57 155535452 EC50 = 852 nM T86679 C67VZK 155535458 Ki > 30000 nM T86679 CI40DC 155535506 Ki > 1000 nM T86679 CV70JY 155536243 IC50 = 2800 nM T86679 C38WUG 155536405 EC50 > 1000 nM T86679 CH6E1O 155536745 Ki = 1.69 nM T86679 C6Q1EM 155536934 Ki > 10000 nM T86679 CMG75B 155537001 Ki > 1000 nM T86679 C8ZG7F 155537023 Ki > 1000 nM T86679 CI5JE0 155537122 IC50 = 56 nM T86679 CSZT95 155537221 Ki = 27.03 nM T86679 C5QUZ2 155537448 IC50 > 10000 nM T86679 CS93VH 155537687 IC50 = 440 nM T86679 CM12WR 155537810 IC50 = 490 nM T86679 CIKT51 155538777 IC50 > 10000 nM T86679 CD9KW3 155539920 Ki > 300 nM T86679 CT7A3I 155540193 Ki > 1000 nM T86679 C4J5VI 155540197 IC50 = 97 nM T86679 C8BHN2 155540525 IC50 > 30000 nM T86679 CF6ZE5 155540615 Ki > 1000 nM T86679 C3P1ZT 155540839 Ki > 1000 nM T86679 CJ4PS8 155540888 Ki > 1000 nM T86679 C2L9TS 155540948 Ki > 1000 nM T86679 C4KDO9 155541051 EC50 = 982 nM T86679 C56VYE 155541183 IC50 = 790 nM T86679 CBE65T 155541185 Ki > 300 nM T86679 C19HQM 155541262 Ki > 1000 nM T86679 CU6F8S 155541364 IC50 = 3400 nM T86679 C2HX6J 155541790 IC50 > 30000 nM T86679 C9H5VC 155541975 Ki > 30000 nM T86679 CQ1FY8 155542311 EC50 > 1000 nM T86679 CMEW36 155542520 EC50 > 1000 nM T86679 CGY1J4 155542588 Ki > 10000 nM T86679 CCV87Q 155542600 Ki > 1000 nM T86679 CNS5H2 155542641 IC50 = 12 nM T86679 C8JY0G 155542643 Ki > 1000 nM T86679 C0BFX9 155542720 Ki = 96.7 nM T86679 C95UDB 155542822 Ki = 731 nM T86679 C06OKY 155542884 IC50 > 30000 nM T86679 CR02FI 155543633 IC50 = 200 nM T86679 C3XDT7 155543719 IC50 > 30000 nM T86679 C2DNQ0 155543871 IC50 > 30000 nM T86679 C1QAZ9 155544096 Ki = 3000 nM T86679 CR0EV6 155544177 IC50 > 30000 nM T86679 CH1G4C 155544368 Ki > 1000 nM T86679 CJHR91 155544551 IC50 = 300 nM T86679 C30NOS 155544777 Ki > 1000 nM T86679 CQ9Z2P 155545386 IC50 > 30000 nM T86679 C5Y4BH 155545414 Ki > 1000 nM T86679 C5HU6A 155545585 Ki = 12.2 nM T86679 C45CUJ 155545762 Ki = 0.352 nM T86679 C2NKO5 155545904 IC50 > 30000 nM T86679 C3B0SI 155546100 IC50 > 30000 nM T86679 C95ICF 155546118 Ki > 10000 nM T86679 C4BHE8 155546183 Ki > 1000 nM T86679 CL1T9K 155546550 IC50 > 30000 nM T86679 C6XP3U 155546562 Ki > 1000 nM T86679 C1X2GS 155546843 Ki > 300 nM T86679 C1VHM5 155547186 IC50 > 30000 nM T86679 CQE30Y 155547305 Ki > 10000 nM T86679 CXAV84 155547390 EC50 > 1000 nM T86679 CK1X5S 155547588 Ki > 1000 nM T86679 C42XEK 155547698 Ki > 1000 nM T86679 C6XJ0D 155547715 EC50 > 1000 nM T86679 C8Q7JG 155547782 Ki > 1000 nM T86679 C7IV9G 155548102 IC50 = 390 nM T86679 CK1BN8 155548182 IC50 = 280 nM T86679 C35WAK 155548264 Ki = 1.91 nM T86679 C39GTQ 155548778 IC50 > 30000 nM T86679 CY1XJ0 155548779 IC50 > 30000 nM T86679 C4MIT2 155548780 Ki > 1000 nM T86679 CF8UJ6 155548797 Ki = 117.8 nM T86679 CYM0W2 155548802 IC50 = 150 nM T86679 C3NE6F 155549264 Ki = 3.55 nM T86679 C6CDL3 155549589 IC50 = 210 nM T86679 CT1Z7V 155549654 IC50 = 97 nM T86679 CC45SE 155550088 Ki > 1000 nM T86679 CY7Q9N 155550159 Ki = 0.153 nM T86679 C4SY8L 155550407 IC50 = 130 nM T86679 C2IU1J 155550532 Ki > 1000 nM T86679 C1Q5BI 155550704 Ki = 238 nM T86679 C6J5EX 155550807 Ki > 1000 nM T86679 CN2I3H 155550832 Ki > 10000 nM T86679 CN5O1L 155551418 IC50 = 540 nM T86679 C5BC3H 155551596 EC50 > 1000 nM T86679 CAO05B 155551709 IC50 = 2.4 nM T86679 C4LN3W 155551750 Ki = 7.02 nM T86679 C6UKR7 155552077 IC50 = 1100 nM T86679 CA29GP 155552390 IC50 > 30000 nM T86679 CJ82KN 155552405 Ki = 5.69 nM T86679 CD26XI 155552481 IC50 = 760 nM T86679 CM40UT 155552539 Ki > 1000 nM T86679 CIQH30 155552719 Ki > 1000 nM T86679 CX7W0G 155552737 EC50 > 1000 nM T86679 CPN79B 155553292 EC50 > 1000 nM T86679 CX4P7S 155553385 Ki > 30000 nM T86679 CD42WK 155553510 IC50 > 30000 nM T86679 CNK6Z9 155553575 Ki = 4.31 nM T86679 C1A5OR 155553697 Ki > 1000 nM T86679 CB75AP 155553750 Ki > 1000 nM T86679 CNGQ04 155553932 IC50 = 8.8 nM T86679 CU1ZE5 155554091 IC50 = 13 nM T86679 CPXQ16 155554464 IC50 = 152 nM T86679 C57MKC 155555241 Ki > 1000 nM T86679 CTHQ10 155555355 IC50 = 190 nM T86679 CVDO87 155555721 Ki = 0.0835 nM T86679 CN38KO 155555854 IC50 > 30000 nM T86679 CL3IB5 155555868 Ki > 10000 nM T86679 CB6XD7 155555919 Ki = 42.1 nM T86679 CJ73SL 155556032 Ki > 1000 nM T86679 CDR63F 155556134 IC50 > 30000 nM T86679 C2VP0T 155556202 Ki > 300 nM T86679 CV9P2M 155556457 Ki > 1000 nM T86679 CC14ON 155556524 Ki > 1000 nM T86679 C1N4WK 155556575 Ki = 234 nM T86679 CNM4F3 155556727 Ki > 1000 nM T86679 C7M1VE 155556836 IC50 > 30000 nM T86679 CGF0H2 155556884 Ki = 1.24 nM T86679 C8QW7M 155556988 Ki > 1000 nM T86679 C9MWG2 155557128 Ki > 1000 nM T86679 CV21NW 155557226 Ki > 1000 nM T86679 CTSX95 155557611 Ki > 1000 nM T86679 CJ16GB 155557960 Ki > 1000 nM T86679 CKA6B3 155558166 IC50 = 260 nM T86679 C7FUQ6 155558172 EC50 > 1000 nM T86679 C0W7AL 155558312 Ki > 1000 nM T86679 CDMC47 155558350 IC50 > 30000 nM T86679 C3A7MK 155558447 Ki > 1000 nM T86679 C8Z2TC 155558489 Ki > 1000 nM T86679 CIAE48 155558941 IC50 > 30000 nM T86679 CVS4T6 155559056 IC50 > 30000 nM T86679 CDZX46 155559070 EC50 > 1000 nM T86679 CTI57G 155559203 Ki > 1000 nM T86679 C2B8NX 155559219 Ki > 300000 nM T86679 CMBE51 155559377 IC50 = 4900 nM T86679 CP87XK 155559423 Ki > 1000 nM T86679 CQM64H 155559636 IC50 > 30000 nM T86679 CG75LM 155559834 IC50 = 73 nM T86679 C34ORN 155560261 IC50 > 30000 nM T86679 C8B7CG 155560391 Ki > 1000 nM T86679 C5X9VL 155560449 Ki = 52.27 nM T86679 C73XYW 155560510 Ki = 0.244 nM T86679 C3OP1F 155560545 Ki > 1000 nM T86679 CN93BY 155560649 EC50 > 1000 nM T86679 CY7BE2 155560676 IC50 = 440 nM T86679 CEXP80 155561009 Ki > 1000 nM T86679 C5KY7D 155561141 Ki = 0.473 nM T86679 CGD7R4 155561189 Ki = 18.6 nM T86679 C1IA4X 155561597 Ki > 1000 nM T86679 CKG56Z 155562044 Ki = 11500 nM T86679 CXUN73 155562096 EC50 > 1000 nM T86679 C6EN2B 155562182 Ki = 4.3 nM T86679 CPDX81 155562247 IC50 = 1500 nM T86679 C30DWF 155562321 Ki = 13.75 nM T86679 C1GHD9 155562338 IC50 = 2300 nM T86679 C1NF2M 155562789 Ki > 1000 nM T86679 CM46KC 155563177 Ki > 1000 nM T86679 CQ19VC 155563189 Ki > 1000 nM T86679 CA27NL 155563199 Ki > 1000 nM T86679 CJZO26 155563438 IC50 > 30000 nM T86679 CPTM25 155563673 Ki > 1000 nM T86679 CG4WA8 155563730 Ki = 651 nM T86679 C5ZKN0 155563788 Ki > 1000 nM T86679 CD6QW7 155563833 Ki > 300 nM T86679 CE2V5Y 155564179 Ki > 1000 nM T86679 C8TL6J 155564465 Ki = 0.643 nM T86679 CHJ5Q8 155564753 IC50 > 30000 nM T86679 CKGC67 155565439 Ki > 300 nM T86679 C0UFM3 155565444 EC50 > 1000 nM T86679 C8N3PQ 155565636 Ki > 1000 nM T86679 CYI54E 155565672 Ki > 1000 nM T86679 CI2CQ0 155565683 Ki > 1000 nM T86679 CB14WJ 155565911 Ki = 8.34 nM T86679 C0VUO9 155566764 Ki = 7.15 nM T86679 CN8RL3 155567003 IC50 > 30000 nM T86679 CCL38W 155568402 IC50 = 1200 nM T86679 C5KNM6 155569051 Ki > 10000 nM T86679 CH86AJ 155569073 Ki > 1000 nM T86679 CH9WE6 155569093 IC50 = 55 nM T86679 C7Q9WY 11395785 EC50 = 16850 nM T86679 C4EBT3 16109359 EC50 = 2041.74 nM T86679 D00ASZ 16204411 EC50 = 2580 nM T86679 D00CJJ 12016636 Ki > 30000 nM T86679 D00GNW 16109429 Ki = 300 nM T86679 D00JWA 46880333 Ki = 7 nM T86679 D00MFV 44572293 Ki = 19000 nM T86679 D01AAI 4046493 Ki = 10000 nM T86679 D01CQU 5139184 Ki = 1.39 nM T86679 D01QBK 44572356 Ki > 30000 nM T86679 D01QYQ 6603931 Ki = 1.9 nM T86679 D01VEU 44300688 IC50 >= 100000 nM T86679 D01VXC 11278089 Ki = 42.5 nM T86679 D01WNA 5248753 Ki = 840 nM T86679 D02HOL 11849871 Ki = 200 nM T86679 D02HYT 11438116 Ki = 76.6 nM T86679 D02JMR 16202727 EC50 = 216 nM T86679 D02RBK 9904551 Ki > 30000 nM T86679 D02RMR 101420 Ki = 1770 nM T86679 D02XPR 73124 Ki > 30000 nM T86679 D03JFX 7 Ki > 30000 nM T86679 D03KKK 169317 Ki = 1110 nM T86679 D03NVE 10226014 Ki = 7 nM T86679 D03RFA 657378 Ki = 43 nM T86679 D04DVT 126079 Ki = 39.81 nM T86679 D04JIR 69689 Ki > 30000 nM T86679 D04LZN 44572409 Ki = 4100 nM T86679 D04WBU 12905388 Ki = 1620 nM T86679 D04WHE 247436 Ki = 1700 nM T86679 D04YUM 75929 Ki > 30000 nM T86679 D05KEF 44418996 Ki = 300 nM T86679 D05XGF 44186581 Ki = 0.393 nM T86679 D06GOE 135465785 Ki = 47 nM T86679 D06GTI 135416058 Ki = 24 nM T86679 D06KYP 44572292 Ki = 1100 nM T86679 D06RCT 16203429 EC50 = 299 nM T86679 D06SGU 11774068 Ki = 6 nM T86679 D06YJN 44459941 Ki = 3390 nM T86679 D07DOE 44447542 Ki = 4440 nM T86679 D07FZA 135522368 Ki = 10 nM T86679 D07HKU 1328 Ki = 62 nM T86679 D07HNM 22995178 Ki = 1330 nM T86679 D08EBT 10981286 EC50 = 100000 nM T86679 D08FOT 5311479 Ki = 53.4 nM T86679 D08FSF 14969716 Ki = 461 nM T86679 D09QLB 1908 Ki = 1330 nM T86679 D09VOP 16203665 EC50 = 1250 nM T86679 D0A0VT 44572291 Ki > 30000 nM T86679 D0A2WH 14969715 Ki = 421 nM T86679 D0A4MK 135489238 Ki = 16 nM T86679 D0A6IO 5310960 Ki = 2056 nM T86679 D0A6JX 452612 Ki = 17000 nM T86679 D0A9BZ 11605883 Ki = 1.33 nM T86679 D0AI8F 12016633 Ki = 860 nM T86679 D0B0TX 44572355 Ki = 4200 nM T86679 D0B1YW 15627855 Ki = 4.7 nM T86679 D0B3NZ 981611 Ki > 1000 nM T86679 D0B3UE 12852 Ki > 30000 nM T86679 D0B9CC 10869347 Ki = 646 nM T86679 D0C1PS 12486289 Ki > 30000 nM T86679 D0C2UJ 8974 Ki = 21400 nM T86679 D0CX7N 44572471 Ki = 5100 nM T86679 D0D9YL 11821203 Ki = 10200 nM T86679 D0DB7A 414707 Ki = 16000 nM T86679 D0E2FV 309375 Ki > 30000 nM T86679 D0E4UT 13789211 Ki > 30000 nM T86679 D0E8RA 2773172 Ki = 7100 nM T86679 D0F4EN 11470612 IC50 > 1000 nM T86679 D0F4XB 2817165 Ki = 34 nM T86679 D0G6BI 16203542 EC50 = 109 nM T86679 D0G6VT 16202726 EC50 = 1870 nM T86679 D0H9BP 5697 Ki = 7.75 nM T86679 D0H9EY 10475082 Ki = 1150 nM T86679 D0HE1P 11717831 EC50 = 31 nM T86679 D0HK5B 9798914 Ki > 10000 nM T86679 D0I1IW 16203539 EC50 = 767 nM T86679 D0IG5E 44582613 Ki = 4830 nM T86679 D0IJ2X 10219753 Ki = 552 nM T86679 D0J4EZ 135443359 Ki = 36 nM T86679 D0JJ6T 10021483 Ki = 4930 nM T86679 D0K0OT 1329 IC50 = 3.8 nM T86679 D0K6ZA 5311041 Ki = 0.4 nM T86679 D0K8ZW 10998551 Ki = 965 nM T86679 D0K8ZZ 448222 EC50 = 3.162 nM T86679 D0L0VU 135484064 Ki = 5.5 nM T86679 D0L6YI 16203540 EC50 = 365 nM T86679 D0L8DZ 12295530 Ki = 810 nM T86679 D0LD0X 128525 Ki = 360 nM T86679 D0M3CG 93205 EC50 = 1680 nM T86679 D0M7AX 10219934 Ki = 4890 nM T86679 D0N8RM 242652 Ki > 30000 nM T86679 D0NO5E 7315331 Ki = 391 nM T86679 D0O0FP 9860294 Ki = 352 nM T86679 D0O1CW 2840092 Ki = 1780 nM T86679 D0O4KI 9834769 Ki = 721 nM T86679 D0O6NS 81457 Ki > 30000 nM T86679 D0OR5V 414708 Ki > 30000 nM T86679 D0P0BV 16202841 EC50 = 896 nM T86679 D0P7FK 743242 Ki = 220 nM T86679 D0P8MK 44572469 Ki = 2800 nM T86679 D0PB2W 1892 Ki = 17300 nM T86679 D0Q1RD 16202725 EC50 = 2180 nM T86679 D0Q6KO 1942 Ki > 30000 nM T86679 D0Q6WX 2690 Ki = 9.8 nM T86679 D0Q9GL 135443367 Ki = 12 nM T86679 D0R1XY 123807 Ki = 42 nM T86679 D0R8OK 822296 Ki = 720 nM T86679 D0RZ5U 101446 Ki = 9490 nM T86679 D0S4JI 20262 Ki > 30000 nM T86679 D0S5XP 44572408 Ki = 4600 nM T86679 D0S6QA 11608719 Ki = 5600 nM T86679 D0T7GG 16109430 Ki = 300 nM T86679 D0TC7N 9953255 EC50 > 100000 nM T86679 D0TU7I 5353365 Ki > 1000 nM T86679 D0U8DW 11781054 Ki = 11.8 nM T86679 D0V2NH 14969717 Ki = 408 nM T86679 D0V7MX 247678 Ki > 30000 nM T86679 D0V8MD 1922 IC50 = 210 nM T86679 D0V9EE 24950370 Ki = 170 nM T86679 D0W1PF 16109428 Ki = 300 nM T86679 D0W6FC 44572473 Ki = 640 nM T86679 D0W6TG 44186666 Ki = 0.157 nM T86679 D0W8RB 44572357 Ki > 30000 nM T86679 D0X5PJ 135529391 Ki = 56 nM T86679 D0Y5TL 5372720 Ki = 3.8 nM T86679 D0Y5WQ 44185871 IC50 = 0.534 nM T86679 D0Y8LD 135529386 Ki = 32 nM T86679 D0Y8SB 4355631 IC50 = 3000 nM T86679 D0Y9WZ 44583036 Ki = 1.2 nM T86679 D0Z1WY 44447548 Ki = 4470 nM T86679 D0Z2QM 23562742 Ki > 30000 nM T86679 D0Z7BC 44442164 Ki > 10000 nM T86679 D0Z8NC 16109435 Ki = 300 nM T86679 D0Z8VU 44572295 Ki = 1200 nM T86679 D0ZF8N 11196622 IC50 > 1000 nM T34949 CPS12B 53317097 IC50 > 30000 nM T34949 CGUA26 57331668 IC50 > 30000 nM T34949 CSE6Z5 71463101 EC50 = 8800 nM T06955 D09GOS 2812 IC50 = 1600 nM T06955 D0K8KX 5280343 IC50 = 10000 nM T06955 D00XBC 46861584 Ki = 10 nM T06955 D0O2XQ 11256587 IC50 > 10000 nM T06955 D0E2QN 23585443 IC50 = 3.981 nM T06955 D0J1FL 10308720 IC50 = 501.19 nM T06955 D0W0LS 183789 IC50 > 10000 nM T06955 CY4WG9 3793 IC50 = 500 nM T06955 CQ3KO7 483339 IC50 > 1000 nM T06955 C7AP9W 483340 IC50 > 1000 nM T06955 CAB79M 483341 IC50 > 1000 nM T06955 C7XW2D 483342 IC50 > 1000 nM T06955 C7PMT6 483343 IC50 > 1000 nM T06955 CP25RI 483344 IC50 > 1000 nM T06955 C71OYP 3758269 IC50 > 25000 nM T06955 CCJ0S5 5071677 IC50 = 900 nM T06955 CMT8K7 5481702 IC50 = 10000 nM T06955 CHCY06 6918496 IC50 > 10000 nM T06955 C8F0RP 9827294 Ki = 0.7943 nM T06955 C9OWM1 9856506 IC50 = 260 nM T06955 C84VKH 9943773 IC50 = 210 nM T06955 C91RTG 9956238 IC50 > 10000 nM T06955 CI9F5T 9959269 Ki = 3.162 nM T06955 CBE6S5 10126022 IC50 = 1258.93 nM T06955 CXVQ60 10133595 IC50 = 45 nM T06955 C49UDP 10150948 IC50 = 125.89 nM T06955 CGA69D 10173173 IC50 = 3162.28 nM T06955 CKH6F8 10193586 IC50 = 39.81 nM T06955 C7CAJ1 10193603 IC50 = 630.96 nM T06955 C5JF6R 10194274 IC50 = 199.53 nM T06955 CM4WK5 10194488 IC50 = 199.53 nM T06955 C8GSV4 10195057 IC50 = 0.631 nM T06955 CC2UA3 10195081 IC50 = 12.59 nM T06955 C56OCZ 10215932 IC50 = 63.1 nM T06955 C3G7DB 10238794 IC50 = 0.3162 nM T06955 CK49NQ 10272003 IC50 > 10000 nM T06955 C1P2OL 10287052 IC50 = 7.943 nM T06955 C43BTO 10287192 IC50 = 39.81 nM T06955 C9NQE8 10287210 IC50 = 125.89 nM T06955 CXPS29 10288569 IC50 = 39.81 nM T06955 C7H4FW 10308962 IC50 = 79.43 nM T06955 C9C6AP 10308963 IC50 = 15.85 nM T06955 CMDA29 10309206 IC50 = 12.59 nM T06955 C0X8QE 10309892 IC50 = 5011.87 nM T06955 CT7GY3 10309893 IC50 = 10 nM T06955 CIL92W 10309983 IC50 = 1000 nM T06955 CWFB30 10323427 IC50 > 2000 nM T06955 CK21LX 11223594 IC50 = 270 nM T06955 C3H8QV 11234202 IC50 = 7.943 nM T06955 C3HO4L 11244702 IC50 = 19.95 nM T06955 C06TUD 11285791 IC50 = 1100 nM T06955 CXL7K1 11496063 IC50 = 31 nM T06955 CUA67M 11525206 Ki = 2.512 nM T06955 C7X3CQ 15604497 Ki = 1995.26 nM T06955 CQJ7Y2 15985912 Ki = 398.11 nM T06955 CDU1L0 16041411 IC50 = 3723 nM T06955 C9G8TZ 16124598 Ki = 794.33 nM T06955 CBM96X 16724339 IC50 = 19 nM T06955 C8BCQ3 16747697 Ki = 100 nM T06955 CES62Q 20299676 IC50 = 280 nM T06955 CMXV34 21866577 IC50 = 37 nM T06955 CZ68SW 21866580 IC50 = 340 nM T06955 CWZ5K1 23585446 IC50 = 3.981 nM T06955 CDCR41 25141190 IC50 = 18 nM T06955 CXFU01 25141301 IC50 = 24 nM T06955 CL3J1C 25212379 IC50 = 19 nM T06955 C84VAR 25212472 IC50 = 30 nM T06955 C54LQF 25230828 IC50 > 50000 nM T06955 C91AYO 36053257 Ki > 29000 nM T06955 CU2PO5 44180522 IC50 > 10000 nM T06955 CXH45J 44288481 IC50 = 9000 nM T06955 CY09MO 44288557 IC50 = 100000 nM T06955 C6OTL1 44288575 IC50 = 7000 nM T06955 CE5U2B 44288633 IC50 ~ 6000 nM T06955 C6LF3M 44288663 IC50 = 570 nM T06955 C8EF6K 44288682 IC50 = 830 nM T06955 C5E1YT 44288683 IC50 = 4000 nM T06955 C14PGO 44288698 IC50 = 7000 nM T06955 CFRD60 44288725 IC50 > 100000 nM T06955 CJX20K 44288726 IC50 = 34000 nM T06955 CQ4BH8 44288730 IC50 = 1000 nM T06955 C3N5GR 44288731 IC50 = 11000 nM T06955 CVYN26 44288732 IC50 = 1000 nM T06955 CTB8K3 44288733 IC50 > 100000 nM T06955 CK14ST 44288776 IC50 = 11000 nM T06955 CLC87J 44288779 IC50 = 33000 nM T06955 CXGE74 44288791 IC50 = 19000 nM T06955 C06TZB 44288799 IC50 = 690 nM T06955 C3OVU9 44288818 IC50 = 830 nM T06955 CTUV63 44288827 IC50 = 18000 nM T06955 CD65QZ 44288828 IC50 = 8000 nM T06955 CIL9Q7 44288854 IC50 = 1000 nM T06955 CM0H9D 44288863 IC50 = 100000 nM T06955 CC8K7V 44288879 IC50 = 2000 nM T06955 CT3NS8 44288880 IC50 = 200 nM T06955 C2DOG1 44288897 IC50 = 5600 nM T06955 C2JAO8 44288898 IC50 = 36000 nM T06955 C1Q0ML 44288899 IC50 = 100000 nM T06955 CZYM61 44288903 IC50 = 310 nM T06955 C7ZV6O 44288904 IC50 = 360 nM T06955 CC8A9B 44288911 IC50 = 2500 nM T06955 C2WV8J 44288912 IC50 = 24000 nM T06955 CQGL52 44288913 IC50 = 1500 nM T06955 CRT26B 44288923 IC50 = 4000 nM T06955 CAX6U8 44288943 IC50 = 1500 nM T06955 C3IJH2 44288958 IC50 = 140 nM T06955 CT3Y4J 44288959 IC50 = 110 nM T06955 CMIR29 44288960 IC50 = 10000 nM T06955 CMU41Y 44288961 IC50 = 11000 nM T06955 C5Y8JR 44288962 IC50 = 11000 nM T06955 C0IR9B 44288963 IC50 = 11000 nM T06955 C6F7TY 44288964 IC50 = 930 nM T06955 CBJ28L 44288972 IC50 = 600 nM T06955 CZM91L 44288978 IC50 = 18000 nM T06955 CN82CD 44288981 IC50 = 1400 nM T06955 CX2Y5V 44288985 IC50 = 11000 nM T06955 CXTA70 44288996 IC50 = 250 nM T06955 C4KI5C 44288998 IC50 = 9000 nM T06955 CM91LD 44289027 IC50 = 330 nM T06955 C53DXA 44289036 IC50 = 33000 nM T06955 C60AZW 44289039 IC50 = 2500 nM T06955 C2JL6Y 44289055 IC50 = 7000 nM T06955 CKE51I 44289057 IC50 = 66000 nM T06955 CJDG24 44289062 IC50 = 1300 nM T06955 C9VZH7 44289063 IC50 = 6000 nM T06955 COKQ32 44289064 IC50 = 13000 nM T06955 CESA31 44289072 IC50 = 12000 nM T06955 C7U1DC 44289082 IC50 = 29000 nM T06955 CNZ1A9 44289083 IC50 > 25000 nM T06955 C27TDH 44289097 IC50 = 6000 nM T06955 C39QRX 44289098 IC50 = 32000 nM T06955 C7S8RE 44289105 IC50 = 2400 nM T06955 CL57CT 44289106 IC50 = 33000 nM T06955 C2ZMR9 44289116 IC50 = 21000 nM T06955 CVF6B3 44289186 IC50 = 2300 nM T06955 C3PEF2 44289203 IC50 = 380 nM T06955 CE2Z6O 44289204 IC50 = 3500 nM T06955 C48RKD 44289205 IC50 = 8000 nM T06955 CW5F7E 44289207 IC50 = 100000 nM T06955 CL72XJ 44289208 IC50 = 20000 nM T06955 CN17JU 44289214 IC50 = 11000 nM T06955 C0YHM2 44289227 IC50 = 360 nM T06955 C59EHT 44289235 IC50 = 3500 nM T06955 C3X1UD 44289241 IC50 = 250 nM T06955 CJXM79 44289242 IC50 = 8000 nM T06955 C1IJ2N 44289275 IC50 = 12000 nM T06955 CO1WT4 44289276 IC50 = 340 nM T06955 C3VH5J 44289277 IC50 = 12000 nM T06955 C6K7SN 44289278 IC50 = 9000 nM T06955 C8VDY4 44289281 IC50 = 6700 nM T06955 CTM89Z 44289282 IC50 = 1000 nM T06955 CG2JY0 44289283 IC50 = 6000 nM T06955 CDLI72 44289340 IC50 = 2500 nM T06955 CD75RK 44289341 IC50 = 400 nM T06955 CY3GC5 44289342 IC50 = 440 nM T06955 C8FH0W 44289343 IC50 = 790 nM T06955 C8NPV7 44289401 IC50 = 2900 nM T06955 CD29AX 44400731 IC50 > 30000 nM T06955 C49TZV 44400735 IC50 > 30000 nM T06955 C45WLQ 44400829 IC50 = 2500 nM T06955 CGS3K6 44400830 IC50 = 10000 nM T06955 CL3FP9 44400833 IC50 = 2000 nM T06955 CID29W 44400839 IC50 > 10000 nM T06955 CFG2W3 44400881 IC50 = 25000 nM T06955 CJOX47 44400899 IC50 = 2400 nM T06955 C6C9VD 44400911 IC50 > 10000 nM T06955 CX0B9L 44400922 IC50 = 25000 nM T06955 C4RU7J 44400947 IC50 = 3000 nM T06955 C51REI 44400993 IC50 > 30000 nM T06955 CJ5ZH7 44401007 IC50 = 2800 nM T06955 CC25KY 44401027 IC50 = 1500 nM T06955 C0K8CZ 44401066 IC50 = 2000 nM T06955 C4U0SC 44401087 IC50 = 8000 nM T06955 C5BG7M 44401090 IC50 > 10000 nM T06955 C2MC7K 44401118 IC50 = 6100 nM T06955 CT6C7D 44401153 IC50 = 9000 nM T06955 C2E8ZO 44406246 IC50 = 5600 nM T06955 CCE2G9 44406247 IC50 = 1200 nM T06955 CRB97O 44406253 IC50 > 10000 nM T06955 C19HLC 44406276 IC50 > 10000 nM T06955 CFR50U 44406277 IC50 > 10000 nM T06955 C4MRZ9 44406282 IC50 = 700 nM T06955 CH46IW 44406293 IC50 > 10000 nM T06955 CN04MT 44406309 IC50 = 300 nM T06955 C3RT2A 44406310 IC50 > 10000 nM T06955 CW2AI7 44406335 IC50 = 1000 nM T06955 C8KGE1 44406338 IC50 = 60 nM T06955 C7FI0K 44406339 IC50 > 10000 nM T06955 C9JW8N 44406351 IC50 > 10000 nM T06955 CQD9B0 44406355 IC50 = 800 nM T06955 CH51AU 44410964 IC50 > 25000 nM T06955 CG7UJ5 44410965 IC50 = 1000 nM T06955 C2HY0G 44410966 IC50 = 800 nM T06955 C3ZW4Y 44411022 IC50 > 25000 nM T06955 CM1RF7 44411033 IC50 = 210 nM T06955 CEM6T0 44411034 IC50 > 25000 nM T06955 CGQT30 44411038 IC50 = 12100 nM T06955 CK2SQ8 44411191 IC50 = 370 nM T06955 C2RWM5 44411236 IC50 > 25000 nM T06955 C47OCQ 44411271 IC50 > 25000 nM T06955 C3EG8M 44411321 IC50 = 14 nM T06955 C2YA7M 44411497 IC50 > 25000 nM T06955 C7M5AC 44430302 IC50 = 2100 nM T06955 C95TXP 44430303 IC50 = 4900 nM T06955 C9H1AD 44430304 IC50 = 1100 nM T06955 C32NAM 44430305 IC50 = 2600 nM T06955 CYZG46 44430306 IC50 = 820 nM T06955 CL4VB1 44430307 IC50 = 830 nM T06955 C9OUM3 44430308 IC50 = 280 nM T06955 C0YB9T 44430309 IC50 = 1910 nM T06955 CRK95G 44430310 IC50 = 500 nM T06955 CB87AM 44430311 IC50 = 140 nM T06955 CTD5N2 44430312 IC50 = 3 nM T06955 C1N5XH 44430313 IC50 = 80 nM T06955 C4J3IV 44430317 IC50 = 3600 nM T06955 CZDA01 44440028 Ki = 4600 nM T06955 C8MP9C 44440029 Ki > 29000 nM T06955 CY4D7T 44440031 Ki = 25000 nM T06955 CYRT46 44440033 Ki > 20000 nM T06955 CEMH36 44440041 Ki = 15000 nM T06955 C6PEH5 44440042 Ki > 29000 nM T06955 CVLJ07 44440043 Ki = 10000 nM T06955 CB38GP 44440044 Ki > 33000 nM T06955 C3E9RI 44440045 Ki = 10000 nM T06955 C0H1CR 44440047 Ki = 26000 nM T06955 C5EJH7 44440048 Ki > 10000 nM T06955 CV0Y6E 44440049 Ki > 10000 nM T06955 CNBJ04 44440051 Ki = 1300 nM T06955 CH7T3E 44440054 Ki = 590 nM T06955 C9E5GJ 44440055 Ki = 620 nM T06955 CI6LW8 44440057 Ki > 10000 nM T06955 CLD64O 44440058 Ki > 10000 nM T06955 C5MQU9 44440059 Ki = 2800 nM T06955 CT3XV5 44440060 Ki > 10000 nM T06955 CH5GC1 44440061 Ki > 10000 nM T06955 CJ6Z9F 44440063 Ki > 10000 nM T06955 CKF3J2 44440065 Ki = 850 nM T06955 CCMT93 44440067 Ki > 10000 nM T06955 CSC82L 44440068 Ki > 10000 nM T06955 CJ6M3F 44440072 Ki = 260 nM T06955 C8O2HF 44440075 Ki = 460 nM T06955 C7MK1B 44440076 Ki = 400 nM T06955 C07HPM 44440077 Ki = 820 nM T06955 CO7A9J 44440079 Ki = 470 nM T06955 C19HPL 44440080 Ki = 530 nM T06955 CDV84L 44440081 Ki = 240 nM T06955 CYWM13 44440083 Ki = 280 nM T06955 C80HEI 44440084 Ki = 420 nM T06955 CPT65M 44440135 Ki = 20200 nM T06955 CT5N4E 44555481 IC50 > 50000 nM T06955 CI4QX8 44561137 IC50 = 260 nM T06955 C0K2SX 44561172 IC50 = 32 nM T06955 C5A7IP 44561217 IC50 = 220 nM T06955 C0QRA4 44561294 IC50 = 18 nM T06955 C8VYW3 44561332 IC50 = 550 nM T06955 CQ72SE 44561333 IC50 = 31 nM T06955 CT2LW7 44561334 IC50 = 13 nM T06955 CIB3P7 44561335 IC50 = 200 nM T06955 CHY0G6 44561363 IC50 = 510 nM T06955 CK98UV 44561561 IC50 = 480 nM T06955 CZ7EP5 44561588 IC50 = 200 nM T06955 CID61F 44562155 IC50 = 25 nM T06955 C8SP0T 44562156 IC50 = 220 nM T06955 CXCW30 44562189 IC50 = 31 nM T06955 C7SKA6 44562190 IC50 = 98 nM T06955 CZNO43 44562191 IC50 = 43 nM T06955 C7HI2W 44562192 IC50 = 61 nM T06955 CM95JL 44562235 IC50 = 550 nM T06955 C3V9TE 44562236 IC50 = 92 nM T06955 CH6BE5 44562237 IC50 = 150 nM T06955 CS4A5Z 44562238 IC50 = 130 nM T06955 CS23FZ 44581042 IC50 = 48 nM T06955 C4DE8G 44581043 IC50 = 100 nM T06955 CP65MD 44581044 IC50 = 52 nM T06955 CP0UN6 44581068 IC50 = 100 nM T06955 C41FJB 44581102 IC50 = 87 nM T06955 CN1E2I 44581103 IC50 = 61 nM T06955 CO07FD 44581121 IC50 = 180 nM T06955 C56TZF 44581122 IC50 > 1000 nM T06955 C8HY2G 45104321 IC50 = 4360 nM T06955 CX79QB 45104422 IC50 = 1570 nM T06955 C5RP0T 45104423 IC50 = 4240 nM T06955 CI6RQ0 45104424 IC50 = 8580 nM T06955 CF67NY 45104425 IC50 = 4360 nM T06955 C96FOD 45104426 IC50 = 6040 nM T06955 CY4S7I 45104427 IC50 = 2560 nM T06955 CW5JQ9 45104523 IC50 = 1320 nM T06955 CVAX51 45104524 IC50 = 539 nM T06955 CQGA14 45104525 IC50 = 6000 nM T06955 C4X9SG 45104526 IC50 = 110 nM T06955 C0PC9G 45104527 IC50 = 1590 nM T06955 CJ16RT 45104633 IC50 = 21.2 nM T06955 CFXE50 45104634 IC50 = 131 nM T06955 CR24SG 45104635 IC50 = 15100 nM T06955 CNK3E0 45104746 IC50 > 10000 nM T06955 C7MA6B 45104747 IC50 = 58500 nM T06955 CKA10J 45104748 IC50 = 31300 nM T06955 CPRX76 45104749 IC50 > 10000 nM T06955 C0L6NA 45104750 IC50 = 775 nM T06955 CY5QK4 45104751 IC50 = 1130 nM T06955 C19XHL 45104752 IC50 = 420 nM T06955 CJ1H9W 45104844 IC50 = 389 nM T06955 CJR14E 45104845 IC50 = 478 nM T06955 CX9EG2 45104846 IC50 = 4760 nM T06955 CRB6U5 45104847 IC50 = 5210 nM T06955 CN1K9D 45104848 IC50 = 1640 nM T06955 CV4WL3 45104849 IC50 = 3120 nM T06955 C2HU6A 45104850 IC50 = 7320 nM T06955 C3FQ9H 45104943 IC50 = 527 nM T06955 CYPI49 45104944 IC50 = 671 nM T06955 C9WQP2 45104945 IC50 = 196 nM T06955 C3BZL7 45104946 IC50 = 1510 nM T06955 CK3N1G 46206137 IC50 > 10000 nM T06955 CR1W9J 46232996 IC50 = 836000 nM T06955 CQVG17 49798349 Ki = 398.11 nM T06955 C62VRQ 49798437 Ki = 1584.89 nM T06955 CY90CD 49798461 Ki = 1258.93 nM T06955 C89OMQ 56848670 IC50 = 398.11 nM T06955 CR5W9K 56848673 IC50 = 398.11 nM T06955 CND81M 56848674 IC50 = 50.12 nM T06955 CG58JC 56849395 IC50 = 15.85 nM T06955 CR09LY 57400127 IC50 > 10000 nM T06955 C0BZ7L 58054368 IC50 = 15.85 nM T06955 CKF6H8 58054384 IC50 = 31.62 nM T06955 CUJR05 58054387 IC50 = 79.43 nM T06955 C41OGB 58054475 IC50 = 25.12 nM T06955 CFQ95L 58054487 IC50 = 416.87 nM T06955 CAR1E3 58054491 Ki = 158.49 nM T06955 C0LM2K 58054516 Ki = 19.95 nM T06955 C73NJX 58054532 IC50 = 79.43 nM T06955 CRD76G 58597374 IC50 = 25.12 nM T06955 C6JKM0 58834906 IC50 = 283.4 nM T06955 C4PWA9 58835024 IC50 = 566.2 nM T06955 CCR4T7 58835217 IC50 > 5000 nM T06955 C9IV3O 59168106 IC50 = 3.981 nM T06955 CIT82Z 59168115 IC50 = 50.12 nM T06955 CL72OZ 59168158 IC50 = 19.95 nM T06955 CKOT31 59168165 IC50 = 3.981 nM T06955 CD93CX 59168178 IC50 = 794.33 nM T06955 C40KRL 59168181 IC50 = 2.512 nM T06955 CZ58EW 59168189 IC50 = 100 nM T06955 CJM4O6 59168213 IC50 = 5011.87 nM T06955 C10ZIB 59168214 IC50 = 12.59 nM T06955 C0XIL3 59455973 Ki = 158.49 nM T06955 CIP2T4 59455974 IC50 = 91.2 nM T06955 C9SW2F 59455975 IC50 = 19.95 nM T06955 CML98I 59455976 IC50 = 6.31 nM T06955 CL68ZY 59455988 IC50 = 15.85 nM T06955 CXDY14 59455990 IC50 = 39.81 nM T06955 CW9G5N 59455992 Ki = 125.89 nM T06955 CGU0T3 59456003 Ki = 39.81 nM T06955 CBC6J8 59456010 IC50 = 31.62 nM T06955 C8ZX5I 59456012 IC50 = 100 nM T06955 CA74OB 59456014 IC50 = 15.85 nM T06955 CR62SI 59456019 IC50 = 12.59 nM T06955 CM9W3Q 59456021 IC50 = 316.23 nM T06955 CI0V1M 59456023 IC50 = 100 nM T06955 CHO7E8 59456026 IC50 = 39.81 nM T06955 CO40YT 59456042 IC50 = 100 nM T06955 CYK5G3 59456050 IC50 = 6.31 nM T06955 CZVR70 59456051 Ki = 15.85 nM T06955 CM0F9U 59456058 IC50 = 15.85 nM T06955 CC87NB 59456067 Ki = 7.943 nM T06955 C4IGS6 59456072 Ki = 251.19 nM T06955 C4B8DA 59456098 IC50 = 79.43 nM T06955 C7FPY8 59456102 Ki = 12.59 nM T06955 C92SJM 59456103 IC50 = 15.85 nM T06955 CW8S1J 59456111 IC50 = 39.81 nM T06955 CJ3DL2 70681287 Ki = 251.19 nM T06955 C1X0JK 70685473 IC50 = 32.36 nM T06955 C1DYW8 70685474 IC50 = 128.82 nM T06955 CYU09C 70689680 Ki = 251.19 nM T06955 CWSU19 70693879 IC50 = 47.86 nM T06955 CG5V6I 71214710 Ki = 630.96 nM T06955 CA72CU 71214725 Ki = 630.96 nM T06955 CMSH09 71214976 Ki = 1000 nM T06955 C24QMP 71449124 IC50 = 4000 nM T06955 CSD6R9 71450657 Ki = 398.11 nM T06955 C8A0XW 71450658 Ki = 158.49 nM T06955 C8YW2L 71452487 Ki = 1258.93 nM T06955 C1TOE8 71452488 Ki = 3981.07 nM T06955 C6PYG7 71452724 IC50 = 20000 nM T06955 C71FXH 71454246 Ki = 501.19 nM T06955 CSL01M 71454248 Ki = 501.19 nM T06955 C6RO2Y 71454500 IC50 = 1200 nM T06955 C3EYK5 71456007 Ki = 3162.28 nM T06955 CHV16Z 71456008 Ki = 3162.28 nM T06955 C6MHX5 71457815 Ki = 1000 nM T06955 CNL64C 71458049 IC50 = 18000 nM T06955 C3BXS9 71461438 Ki = 2511.89 nM T06955 CRV73F 71461439 Ki = 1258.93 nM T06955 C3P5HM 71461440 Ki = 2511.89 nM T06955 CB4OJ1 71461546 IC50 = 110 nM T06955 C0LT6D 71461653 IC50 = 17000 nM T06955 C3B2XY 71462571 Ki = 10 nM T06955 C5E1FJ 71463165 Ki > 10000 nM T06955 C8VX0L 71463166 Ki > 10000 nM T06955 C6Y4KW 71583039 IC50 = 251.19 nM T06955 CDK4U2 71583488 IC50 = 19.95 nM T06955 CX26AC 71583489 IC50 = 31.62 nM T06955 CBGO13 71583704 IC50 = 251.19 nM T06955 CYEU10 71584535 IC50 = 158.49 nM T06955 CL94NI 71584536 IC50 = 100 nM T06955 C1DWU2 71584537 IC50 = 125.89 nM T06955 CZG2O3 71720517 IC50 = 9900 nM T06955 C6ENV5 100951623 EC50 > 10000 nM T06955 CI9DP8 118706816 IC50 = 602.56 nM T06955 CQ4DH6 118706818 IC50 = 199.53 nM T06955 CKT2J4 118706819 IC50 = 19952.62 nM T06955 CIA46Y 118706820 IC50 = 1995.26 nM T06955 C14FQW 118706821 IC50 = 457.09 nM T06955 CN9O1I 118706822 IC50 > 31622.78 nM T06955 C2B4YR 118706823 IC50 = 1000 nM T06955 CXB1D5 118706824 IC50 = 112.2 nM T06955 C2YTI5 118706825 IC50 = 3981.07 nM T06955 CTP74U 118706826 IC50 = 1995.26 nM T06955 CV24FW 118706827 IC50 = 1584.89 nM T06955 COD3W0 118706828 IC50 = 398.11 nM T06955 CRI37O 118706829 IC50 = 199.53 nM T06955 CB4EX3 127045756 Ki = 1.585 nM T06955 CXJU02 127045975 Ki = 25.12 nM T06955 C63YVS 127045976 Ki = 15.85 nM T06955 COI4B9 127045977 Ki = 100 nM T06955 CBW04F 127045978 Ki = 25.12 nM T06955 C4PF8W 127046189 Ki = 19.95 nM T06955 CPGL57 127046190 Ki = 50.12 nM T06955 CK4RX7 127046247 Ki = 2.512 nM T06955 CC4W0D 127046612 Ki = 3.981 nM T06955 CZ86TM 127046613 Ki = 25.12 nM T06955 CU3Y0X 127046614 Ki = 3.162 nM T06955 CPH5I2 127046787 Ki = 25.12 nM T06955 C40MAY 127047356 Ki = 1 nM T06955 C7RHL4 127047440 EC50 = 398.11 nM T06955 CF4I1Q 127047441 Ki = 316.23 nM T06955 C38GVH 127047612 Ki = 5.012 nM T06955 CUR0S2 127047970 Ki = 50.12 nM T06955 C5ZX4A 127047971 Ki = 125.89 nM T06955 CMG47H 127047972 Ki = 630.96 nM T06955 C4AC6W 127047973 Ki = 100 nM T06955 CN50EP 134324770 IC50 = 638 nM T06955 CQ8O4F 134324821 IC50 = 228 nM T06955 CRD52S 134324842 IC50 = 40 nM T06955 CYG68S 134324891 IC50 = 58 nM T06955 CG4VU0 134324973 IC50 = 47 nM T06955 CA7NV8 134324996 IC50 = 837 nM T06955 CEH7V6 134325003 IC50 = 37 nM T06955 C17NBC 134325016 IC50 = 27 nM T06955 C2LJ5X 134325041 IC50 = 32 nM T06955 CHWL68 134325076 IC50 = 32 nM T06955 CYLD56 134325106 IC50 = 23 nM T06955 C51ZNK 134325169 IC50 = 238 nM T06955 C3IP6E 134325215 IC50 = 69 nM T06955 CW7SZ2 134325269 IC50 = 670 nM T06955 C87DJK 134325276 IC50 = 172 nM T06955 C7EP5J 134335265 IC50 = 251 nM T06955 CI85WX 134335393 IC50 = 36 nM T06955 CI5TO1 134335394 IC50 = 34 nM T06955 C03HJQ 136116031 IC50 = 12.59 nM T06955 CT6K3M 137632086 IC50 = 630.96 nM T06955 CH97WT 137632304 IC50 = 794.33 nM T06955 C18RMP 137632634 IC50 = 12589.25 nM T06955 C5S0TY 137632888 IC50 = 316.23 nM T06955 C43HNM 137632974 IC50 = 3162.28 nM T06955 CLMV26 137633709 IC50 = 158.49 nM T06955 CS9NK5 137634526 IC50 = 794.33 nM T06955 CEN4A2 137636457 IC50 > 31622.78 nM T06955 C0O8PZ 137636569 IC50 = 63.1 nM T06955 CKB83H 137637450 IC50 = 7943.28 nM T06955 CMVH92 137638825 IC50 = 501.19 nM T06955 CMW37P 137639432 IC50 = 79.43 nM T06955 CYA6X9 137639968 IC50 = 79.43 nM T06955 C7F4IZ 137642528 IC50 = 10000 nM T06955 C1N6VU 137643503 IC50 = 15848.93 nM T06955 CY03MP 137643926 IC50 = 199.53 nM T06955 C4EQ5T 137644457 IC50 = 316.23 nM T06955 CEM2C5 137644970 IC50 = 794.33 nM T06955 C3WS4U 137645516 IC50 > 31622.78 nM T06955 C8OU7T 137647817 IC50 = 251.19 nM T06955 CH0K3A 137647898 IC50 = 794.33 nM T06955 C9J0KG 137652382 IC50 = 3162.28 nM T06955 CE7PR5 137652824 IC50 = 1258.93 nM T06955 CUF9E8 137652889 IC50 = 630.96 nM T06955 CZC5V3 137653647 IC50 = 251.19 nM T06955 C7HOM5 137654717 IC50 = 630.96 nM T06955 CK3W1Z 137656805 IC50 = 3981.07 nM T06955 C25WIF 137659242 IC50 = 10000 nM T06955 CT18FM 137661320 IC50 = 1995.26 nM T06955 CO4UJ0 137661613 IC50 = 251.19 nM T06955 C14OBI 142450222 IC50 = 275 nM T06955 CK5C4E 145949792 IC50 = 1000 nM T06955 C2MO3X 145950145 IC50 = 3162.28 nM T06955 C3IKC5 145950218 IC50 = 3162.28 nM T06955 C7B5CI 145951136 IC50 = 63.1 nM T06955 C53TWM 145951247 IC50 = 630.96 nM T06955 CW4KT0 145951541 IC50 = 15.85 nM T06955 C3TW7M 145953370 IC50 > 10000 nM T06955 CV9BJ5 145955299 IC50 = 10000 nM T06955 CR92JH 145955410 IC50 = 5011.87 nM T06955 CM06VB 145955548 IC50 = 7943.28 nM T06955 CFY7L3 145955692 IC50 = 158.49 nM T06955 CI8XO5 145958908 IC50 = 63.1 nM T06955 C9CLW4 145959198 IC50 = 1 nM T06955 C0XY4Q 145971718 IC50 = 158.49 nM T06955 CYD40K 155518637 IC50 = 2580 nM T06955 C5OIR9 155520262 IC50 = 104 nM T06955 CYC38R 155527411 IC50 > 5000 nM T06955 CN4A0O 155531126 IC50 = 42 nM T06955 CCAK28 155540774 IC50 = 1380 nM T06955 CR6S2U 155541406 IC50 = 41 nM T06955 CZ6Y5S 155543069 IC50 = 54 nM T06955 C1VU7R 155543648 IC50 = 126 nM T06955 CB4X3V 155548141 IC50 = 803 nM T06955 COFT70 155557193 IC50 = 1200 nM T06955 C6FUA1 155561858 IC50 = 170 nM T06955 D01RGG 21866574 IC50 = 490 nM T06955 D03VIS 9899450 IC50 = 4500 nM T06955 D06AJH 692856 IC50 = 3000 nM T06955 D06MBD 11176403 IC50 < 3000 nM T06955 D0B3JB 44411037 IC50 = 80 nM T06955 D0CX7I 44411325 IC50 = 2000 nM T06955 D0EV1I 44561260 IC50 = 13 nM T06955 D0G6NY 9814340 IC50 = 80 nM T06955 D0K2UA 44411266 IC50 = 440 nM T06955 D0M7HQ 9814022 IC50 = 170 nM T06955 D0U7FE 9900444 IC50 = 300 nM T06955 D0W1VL 4015979 IC50 = 5500 nM T06955 D0W5OM 44411322 IC50 = 900 nM T06955 D0W6GE 9922232 IC50 = 220 nM T06955 D0ZE9M 44411492 IC50 = 1500 nM T77913 D00JVR 2267 Ki = 1.202 nM T77913 D00NAX 4926 IC50 = 2454.71 nM T77913 D01AZG 5073 Ki = 2.6 nM T77913 D01FGR 3100 Ki = 14.79 nM T77913 D01GBY 124087 Ki = 0.97 nM T77913 D01JUF 5775 IC50 = 316227.77 nM T77913 D01KPV 3348 Ki = 27 nM T77913 D01ZII 2726 Ki = 4.25 nM T77913 D03KQF 4011 Ki = 1.67 nM T77913 D03WEX 9966051 Ki = 180 nM T77913 D04USC 774 EC50 = 13 nM T77913 D05DVP 5717 IC50 > 10000 nM T77913 D05ZIK 4205 Ki = 1.6 nM T77913 D06ABF 3957 Ki = 37 nM T77913 D06MAJ 65906 Ki = 2.7 nM T77913 D06ZUK 3696 IC50 = 27 nM T77913 D08CTT 21855 Ki = 0.6918 nM T77913 D08JZS 4992 IC50 = 0.014 nM T77913 D08VRO 3822 Ki = 2 nM T77913 D0B0CP 667467 Ki = 3.75 nM T77913 D0B4JQ 5587 IC50 = 39.81 nM T77913 D0B7NG 2725 Ki = 0.92 nM T77913 D0CQ0Z 33630 Ki = 1000 nM T77913 D0D1AL 3559 Ki = 440 nM T77913 D0D9FV 4601 IC50 = 97723.72 nM T77913 D0DK8V 2678 Ki = 5.89 nM T77913 D0E1WI 3345 IC50 = 147910.84 nM T77913 D0E8CI 5282443 Ki = 1.6 nM T77913 D0H3HM 60795 Ki = 25.1 nM T77913 D0H7KF 5002 Ki = 8.7 nM T77913 D0I0DL 3689 IC50 = 1000 nM T77913 D0M8PW 9955977 Ki = 50 nM T77913 D0O6SX 3658 Ki = 2 nM T77913 D0P5SA 3372 Ki = 40 nM T77913 D0R1JV 60854 Ki = 5.3 nM T77913 D0R1WR 4919 IC50 = 17782.79 nM T77913 D0R6RO 4184 Ki = 1.7 nM T77913 D0S1CQ 133017 IC50 = 3.9 nM T77913 D0T2XU 4927 IC50 = 5.4 nM T77913 D0T6QX 5736 Ki = 0.62 nM T77913 D0V4QS 135398745 Ki = 1.2 nM T77913 D0Y5UG 2160 Ki = 1.12 nM T77913 D0YG7M 3827 Ki = 0.1585 nM T77913 D0Z1RV 135398737 Ki = 1 nM T77913 D01UUD 9948102 Ki = 1148.15 nM T77913 D07YGH 9976892 Ki = 2511.89 nM T77913 D0C2HI 60680 IC50 = 100 nM T77913 D0E8ZY 9842252 Ki = 19 nM T77913 D0HZ2E 5311271 Ki = 1000 nM T77913 D0LI1C 44469321 IC50 > 10000 nM T77913 D0M9RQ 11697697 IC50 > 10000 nM T77913 D0N1HW 5311200 Ki > 10000 nM T77913 D0OW9L 11973780 IC50 > 10000 nM T77913 D01RAE 133079 Ki > 1600 nM T77913 D02KAF 10103168 EC50 > 0.0001 nM T77913 D03SXN 104943 IC50 ~ 10000 nM T77913 D05FYA 3035905 Ki > 10000 nM T77913 D06DZI 107780 Ki > 10000 nM T77913 D08SOF 5405 IC50 = 1 nM T77913 D09RGW 11753159 Ki = 31.62 nM T77913 D0B4TT 17747460 Ki = 10 nM T77913 D0K9JP 9928332 Ki > 1000 nM T77913 D0M7LV 5761 Ki = 1540 nM T77913 D0OS6O 60149 Ki = 0.51 nM T77913 D0Y2HR 2247 Ki = 2.089 nM T77913 D0Y6SN 5311096 Ki = 630.96 nM T77913 C8D9QE 2031 IC50 = 112201.85 nM T77913 CJ0B9F 3158 Ki = 0.1778 nM T77913 C5H9CN 9287 Ki > 10000 nM T77913 CTQR73 18878 Ki = 3981.07 nM T77913 CFGH18 27620 Ki = 86.3 nM T77913 C2VQH8 29298 Ki = 7696 nM T77913 CNZD18 36381 Ki > 10000 nM T77913 C20AYU 153996 IC50 = 3 nM T77913 CUO7A3 203096 Ki = 0.2512 nM T77913 CYP7U8 409544 Ki = 275.42 nM T77913 C7D4WL 550981 Ki = 6309.57 nM T77913 CKR2N7 621659 IC50 = 160 nM T77913 CGY6C5 647957 Ki < 10000 nM T77913 CB73XL 649745 Ki = 1905.46 nM T77913 C17XTV 652557 Ki = 0.8 nM T77913 C3LU7J 736282 IC50 = 44668.36 nM T77913 CZN6S9 743974 IC50 > 39810.72 nM T77913 C8Q9BF 747187 Ki > 10000 nM T77913 C9EGO2 763018 Ki < 10000 nM T77913 CXD4H9 867637 Ki = 10715.19 nM T77913 C9DWE5 873049 Ki = 4168.69 nM T77913 C89DBR 1072350 Ki = 2630.27 nM T77913 C1YED3 2199935 Ki = 794.33 nM T77913 CST14K 2421311 Ki = 8128.31 nM T77913 C0BD6K 2537688 Ki = 707.95 nM T77913 CX85VC 2581635 Ki > 10000 nM T77913 CPI2C5 2775690 Ki = 399 nM T77913 CAM7I6 3041343 Ki = 6165.95 nM T77913 C6Z4QI 3050372 Ki = 67.9 nM T77913 C5NA6S 3069135 Ki = 62.9 nM T77913 CL3BA9 3201696 IC50 > 20000 nM T77913 C07ORP 3300652 Ki = 426.58 nM T77913 CJ6D8N 3342390 Ki < 1000 nM T77913 C4WJN8 3359700 Ki = 12.59 nM T77913 C7YQD3 3519055 Ki > 10000 nM T77913 C15ZFL 3570228 Ki = 10964.78 nM T77913 CL20WJ 4440801 Ki = 5370.32 nM T77913 C4X7RJ 5282408 IC50 = 1 nM T77913 CSEH41 5310982 EC50 = 251.19 nM T77913 CSM9T8 6603950 Ki = 12 nM T77913 CFN7L4 6604866 Ki = 69.18 nM T77913 CPR2E4 9549064 Ki = 311 nM T77913 C24GNE 9798145 Ki = 1995.26 nM T77913 C8XGV3 9804849 IC50 > 10000 nM T77913 C5Z2KM 9805944 Ki = 4.2 nM T77913 CIH80R 9818650 Ki = 4085 nM T77913 C0AU9L 9826801 Ki = 500 nM T77913 C6KJ7P 9827677 Ki = 58 nM T77913 CI3GE1 9832306 IC50 = 6.8 nM T77913 CBN06W 9839050 Ki = 0.43 nM T77913 CWTA61 9839081 Ki = 0.64 nM T77913 CNB65K 9848303 Ki = 1500 nM T77913 CJ8LT7 9848518 IC50 > 10000 nM T77913 C28IUE 9850828 Ki = 3.63 nM T77913 CT5M1L 9851785 Ki = 890 nM T77913 CK7FJ6 9870185 Ki = 3.981 nM T77913 CF7M2Y 9870460 Ki = 50 nM T77913 CT2C6K 9870702 IC50 > 10000 nM T77913 C2TUG6 9872445 Ki = 19 nM T77913 C34AHG 9880208 Ki = 4466.84 nM T77913 CDLB96 9889149 IC50 > 1000 nM T77913 CFI97S 9904205 IC50 = 6.761 nM T77913 CUN81Q 9905249 Ki > 10000 nM T77913 CYWQ50 9906447 Ki = 5440 nM T77913 C7JFZ5 9906978 Ki = 259.6 nM T77913 CNI49H 9913604 Ki = 150 nM T77913 CF4VO1 9914506 Ki = 15.85 nM T77913 C6F8RG 9918576 IC50 = 309 nM T77913 CWQ75J 9923147 Ki = 13803.84 nM T77913 CI3V0F 9923186 Ki = 5623.41 nM T77913 CAQ52T 9932698 Ki = 64 nM T77913 C4L1GA 9934033 IC50 = 150 nM T77913 CA0B8C 9944610 Ki > 10000 nM T77913 C2PAC8 9958732 Ki = 305 nM T77913 CCO7G5 9971374 Ki = 1258.93 nM T77913 CD5MI4 9979272 Ki = 8.913 nM T77913 C3YB9L 10003483 Ki = 6600 nM T77913 CZW1M7 10005242 Ki = 50.12 nM T77913 C1XK9Y 10019102 IC50 > 10000 nM T77913 CV7R9F 10020040 Ki > 10000 nM T77913 C2JZL1 10048222 IC50 > 1000 nM T77913 CL98OS 10051425 Ki = 550 nM T77913 CMUW84 10064805 Ki = 1000 nM T77913 C4PCO3 10065083 Ki = 911.8 nM T77913 CK38NM 10065106 Ki > 1995.26 nM T77913 C9OQ2S 10066369 Ki = 218.78 nM T77913 CU78GI 10067368 Ki = 1000 nM T77913 CP08FW 10069595 Ki = 354.81 nM T77913 C4Y1OZ 10069660 Ki = 5.012 nM T77913 CCS5V6 10070478 Ki = 7.586 nM T77913 C54EYD 10108561 IC50 < 1000 nM T77913 CX0VB7 10121390 IC50 = 500 nM T77913 CPL92W 10122529 IC50 = 6.42 nM T77913 CX91IM 10123040 IC50 = 4.47 nM T77913 C4LMJ8 10123138 IC50 = 6.69 nM T77913 C7YM5L 10143016 Ki = 50.12 nM T77913 CEZ23W 10147107 IC50 = 6.36 nM T77913 CGLD53 10147218 IC50 = 6.02 nM T77913 CLW3J6 10151756 Ki = 63.1 nM T77913 C5FZA0 10168749 IC50 = 6.53 nM T77913 C17JMY 10169609 IC50 = 6.02 nM T77913 C2PZF9 10177985 Ki = 7 nM T77913 CJ60XT 10190056 IC50 = 6.62 nM T77913 CBZK69 10190413 IC50 = 6.3 nM T77913 C52GAK 10190638 IC50 = 6.59 nM T77913 CSHR17 10190770 IC50 = 6.55 nM T77913 CKX05J 10190842 IC50 = 994 nM T77913 CPA96J 10212223 IC50 = 6.63 nM T77913 CLM81T 10212645 IC50 = 9447 nM T77913 C75BMN 10212725 IC50 = 4.56 nM T77913 CP1FL9 10233656 IC50 = 6.44 nM T77913 C1J2CL 10234086 IC50 = 5.93 nM T77913 CVF1E5 10246054 IC50 = 16.98 nM T77913 C10TFN 10263017 IC50 = 501.19 nM T77913 CHM93N 10264715 IC50 = 398.11 nM T77913 CHLG27 10266140 Ki > 2511.89 nM T77913 CH31DX 10267394 Ki > 10000 nM T77913 CS6MU7 10268636 Ki = 3715.35 nM T77913 CU8Q2K 10283765 IC50 = 6.6 nM T77913 CI3O7X 10283825 IC50 = 436 nM T77913 C60VRF 10284042 IC50 = 6.26 nM T77913 CZNP37 10300214 IC50 = 5011.87 nM T77913 C76SEC 10305069 IC50 = 5.71 nM T77913 CA38EI 10305888 IC50 = 5 nM T77913 CU89JD 10314060 Ki > 10000 nM T77913 C2Y7PR 10315110 Ki = 0.4169 nM T77913 CZ60AJ 10333104 Ki = 0.5 nM T77913 CN1Y6Z 10341609 Ki = 524.81 nM T77913 CGOE95 10343536 Ki = 5900 nM T77913 C63RGN 10347051 Ki = 295 nM T77913 CN8PA7 10357986 IC50 > 10000 nM T77913 CDAC63 10381889 IC50 = 2.344 nM T77913 C69KIB 10385855 IC50 > 10000 nM T77913 C85OHE 10399921 Ki = 3 nM T77913 C5F4WP 10403711 Ki = 7880 nM T77913 CY0U1B 10408773 Ki = 7.943 nM T77913 CZX92O 10420190 IC50 = 3162.28 nM T77913 CI0LK6 10429386 Ki = 1995.26 nM T77913 CIQ02H 10436842 Ki = 398 nM T77913 C70ZTF 10451094 Ki = 28183.83 nM T77913 CM8PV0 10455457 Ki = 4168.69 nM T77913 C1T7QW 10456093 Ki = 203 nM T77913 CRM27I 10472082 Ki = 562.34 nM T77913 COV85C 10472143 Ki = 2500 nM T77913 CI7D9Z 10473209 Ki = 1584.89 nM T77913 CEF2O6 10478367 Ki > 10000 nM T77913 C43ACT 10575070 Ki = 223.87 nM T77913 CRI50E 10885636 IC50 = 795 nM T77913 CD4O9R 10890691 IC50 = 1258.93 nM T77913 CB1HY3 10894144 IC50 = 280 nM T77913 CX65PW 10907460 IC50 = 1820 nM T77913 C4SBO9 10915140 IC50 = 8000 nM T77913 CNB39C 10947658 Ki = 500 nM T77913 C4WV8L 10969390 Ki = 7.244 nM T77913 CF15CY 10986211 EC50 > 0.0001 nM T77913 CJC9K4 11005810 IC50 = 454 nM T77913 CG41BK 11071079 IC50 = 1280 nM T77913 CO81WF 11094685 EC50 > 0.0001 nM T77913 C7DE0U 11113605 IC50 = 1660 nM T77913 CWE5L2 11116130 EC50 > 0.0001 nM T77913 CVE8T3 11121216 Ki = 1400 nM T77913 CUF10O 11126319 EC50 > 0.0001 nM T77913 C0W4SM 11186523 Ki = 1.4 nM T77913 C75RHS 11230427 IC50 = 630.96 nM T77913 C40ZXD 11230971 Ki = 22 nM T77913 CEZ8Q9 11231249 IC50 = 398.11 nM T77913 CC71TB 11241807 IC50 = 2511.89 nM T77913 C82JRU 11253315 IC50 = 2511.89 nM T77913 C46LPF 11264275 IC50 = 1995.26 nM T77913 C92CYH 11265950 Ki = 4 nM T77913 CS1XJ3 11277528 Ki = 12 nM T77913 CY3B9M 11288570 IC50 = 1258.93 nM T77913 CJS9C0 11304851 IC50 > 10000 nM T77913 C5K7JT 11333854 IC50 = 251.19 nM T77913 C98LOU 11346501 IC50 = 1995.26 nM T77913 CC13FL 11349921 IC50 > 10000 nM T77913 CYEV13 11358657 IC50 = 3981.07 nM T77913 CQW25D 11376787 Ki = 5.89 nM T77913 C5ZHK8 11393516 Ki = 3890.45 nM T77913 C85LYP 11430418 IC50 = 1000 nM T77913 CG58SO 11444350 Ki = 158.49 nM T77913 CL0W9D 11459394 IC50 = 1000 nM T77913 C1O9XD 11493620 Ki = 13 nM T77913 CPX26I 11496746 Ki > 3162.28 nM T77913 C5Z7GQ 11497411 Ki > 1995.26 nM T77913 C9YU1O 11497679 Ki = 3981.07 nM T77913 CQT5U8 11497680 Ki = 501.19 nM T77913 C9JD4N 11497924 Ki > 1995.26 nM T77913 C69AMJ 11500781 Ki = 9.3 nM T77913 C3ROH5 11504077 Ki = 1584.89 nM T77913 CLPO39 11508317 IC50 = 6100 nM T77913 COT4H9 11511117 Ki > 3981.07 nM T77913 CDQ18N 11515125 Ki = 79000 nM T77913 CP9RB7 11515387 Ki = 0.8 nM T77913 CZ3D5Y 11518933 Ki > 1995.26 nM T77913 C0WU7G 11518972 Ki = 630.96 nM T77913 CM4B3J 11519133 Ki = 501.19 nM T77913 C08JSL 11519134 Ki > 1258.93 nM T77913 CTNX29 11526451 Ki > 3162.28 nM T77913 CR9NA7 11526531 Ki > 1584.89 nM T77913 CNL15V 11527195 Ki = 1000 nM T77913 C0BC6Y 11530223 Ki = 59 nM T77913 CKI40W 11533362 Ki = 2511.89 nM T77913 CJF92G 11533429 Ki > 3981.07 nM T77913 C2EQ1U 11533448 Ki < 3162.28 nM T77913 C4LOQ9 11533473 Ki = 1584.89 nM T77913 CZW9U3 11534726 Ki > 501.19 nM T77913 C8GZ1I 11539020 IC50 > 10000 nM T77913 CQ08DH 11539632 IC50 = 3.5 nM T77913 CSN91H 11539722 Ki > 3162.28 nM T77913 C0X6CJ 11540474 Ki < 3162.28 nM T77913 C0ZF8J 11544156 Ki = 11 nM T77913 C9UG2V 11544758 Ki > 4000 nM T77913 C5ZY6N 11545813 Ki = 1014 nM T77913 CD14OF 11547466 Ki > 3162.28 nM T77913 C61LDE 11548217 Ki > 2511.89 nM T77913 CKZ9B0 11548239 Ki = 398.11 nM T77913 CPA7K8 11548755 Ki = 2511.89 nM T77913 C34JAV 11551351 IC50 = 256000 nM T77913 C3Y4GR 11555971 Ki > 3162.28 nM T77913 CX1VD8 11562113 Ki > 2511.89 nM T77913 C0JU9T 11562199 Ki < 1995.26 nM T77913 C4N8JS 11562200 Ki > 1995.26 nM T77913 C52PDV 11568714 Ki = 1584.89 nM T77913 CU6EY8 11569996 Ki = 630.96 nM T77913 CASH81 11576387 Ki > 2511.89 nM T77913 C8YLD3 11577158 Ki = 251.19 nM T77913 CR8E2F 11578028 Ki > 2511.89 nM T77913 CXP2M0 11580426 Ki = 12 nM T77913 CW7G3X 11580427 Ki = 4 nM T77913 CE0U8J 11581337 IC50 > 10000 nM T77913 C6D1MA 11584660 Ki = 794.33 nM T77913 CN5DQ9 11585034 Ki > 1258.93 nM T77913 C73UHS 11585248 Ki = 1995.26 nM T77913 CC75MD 11590828 Ki > 3162.28 nM T77913 CYX50J 11591601 Ki = 125.89 nM T77913 CIUL60 11591633 Ki > 3162.28 nM T77913 C9DI6R 11606176 Ki > 3162.28 nM T77913 CO1A5Z 11606378 Ki = 1584.89 nM T77913 CL04ZJ 11606435 Ki > 1584.89 nM T77913 CJC5N8 11606456 Ki > 2511.89 nM T77913 CT16JP 11613587 Ki > 2511.89 nM T77913 CN91SZ 11613873 Ki > 3162.28 nM T77913 CKB59U 11620847 Ki > 1995.26 nM T77913 CXY07A 11621352 Ki = 1995.26 nM T77913 C79OMR 11623756 Ki = 10000 nM T77913 CSB9O5 11623845 Ki = 35 nM T77913 C9FSA8 11627847 Ki > 3162.28 nM T77913 C51IBH 11627879 Ki = 251.19 nM T77913 CE8W1Z 11628452 Ki > 2511.89 nM T77913 CFJN71 11628631 Ki > 2511.89 nM T77913 C0G6PN 11632103 IC50 > 10000 nM T77913 C23XSL 11638166 IC50 = 23000 nM T77913 C0XC2N 11641596 Ki = 2511.89 nM T77913 C25KGE 11641641 Ki = 1258.93 nM T77913 C8DXS0 11642163 Ki = 1000 nM T77913 CYQB50 11648990 Ki = 100 nM T77913 C1HDM5 11653679 Ki = 188.6 nM T77913 C48HCV 11656243 Ki < 794.33 nM T77913 CPE83G 11656848 Ki > 1995.26 nM T77913 CT14BC 11657494 Ki = 1258.93 nM T77913 C2J9IM 11659397 Ki = 75 nM T77913 CH3N1I 11659592 IC50 = 3500 nM T77913 CEL15N 11662194 Ki > 3162.28 nM T77913 CBU0L8 11663504 Ki > 1995.26 nM T77913 C69RQX 11663526 Ki = 1000 nM T77913 C3SJO5 11663578 Ki < 3162.28 nM T77913 C16UWH 11664328 Ki > 1995.26 nM T77913 CNE2K5 11669953 Ki = 1995.26 nM T77913 CWQ3M4 11677768 Ki = 1995.26 nM T77913 C7JVX2 11681378 Ki = 69 nM T77913 C1ZD6V 11685267 Ki > 3162.28 nM T77913 CY36RI 11688223 Ki = 2.1 nM T77913 CG13YQ 11691697 Ki < 2511.89 nM T77913 CE1KI3 11692214 Ki > 1995.26 nM T77913 CGM36K 11692376 Ki > 2511.89 nM T77913 C7Z0SX 11695591 Ki = 1.7 nM T77913 CP3G0Q 11695811 Ki = 2.9 nM T77913 CT5J9M 11699340 Ki > 2511.89 nM T77913 CFCB20 11699532 Ki < 1995.26 nM T77913 CBDC74 11702114 Ki = 1.4 nM T77913 CQ5P2F 11702115 Ki = 1.7 nM T77913 CXFK83 11702578 Ki = 390 nM T77913 CGD80W 11705119 Ki < 3162.28 nM T77913 C78GTN 11709314 Ki = 1000 nM T77913 CN8FE3 11712044 Ki > 2511.89 nM T77913 CXUM63 11720838 Ki > 5011.87 nM T77913 C37DMH 11721190 Ki = 1000 nM T77913 C7PVL8 11730467 IC50 = 1930 nM T77913 CP49IH 11742610 Ki = 12.88 nM T77913 CW3GA7 11759212 Ki = 0.8128 nM T77913 CMDT64 11804748 EC50 > 0.0001 nM T77913 CT4F2C 11808040 Ki = 28.84 nM T77913 CN9M8E 11811722 IC50 = 496 nM T77913 CO2R6A 11816882 IC50 = 7943.28 nM T77913 C4JIZ5 11829635 EC50 > 0.0001 nM T77913 C0X7FJ 11846300 EC50 = 6.761 nM T77913 CAD8P9 11848624 Ki = 624 nM T77913 CM49QW 11848625 Ki = 3600 nM T77913 CCT5G7 11848677 Ki = 520 nM T77913 CMR10F 11848679 Ki = 2600 nM T77913 CXLW54 11948707 Ki = 839 nM T77913 C8JQL7 11957735 IC50 > 10000 nM T77913 CBV2X0 11963995 Ki = 270 nM T77913 C1A2IB 12001199 Ki < 2511.89 nM T77913 CNO57E 12001832 Ki = 31.62 nM T77913 CJ8K3O 12016525 Ki = 53703.18 nM T77913 CNY71B 12192007 Ki = 10715.19 nM T77913 CYU4P5 12739458 Ki < 10000 nM T77913 C28QEX 12765746 Ki = 15 nM T77913 CL6QH3 12914583 Ki > 10000 nM T77913 CB9G2Y 12992627 Ki = 14 nM T77913 CWOJ46 12992629 Ki = 50 nM T77913 C2V9FL 13091268 Ki = 8780 nM T77913 C2VAE5 13091273 Ki = 635.4 nM T77913 CCG14E 13091356 Ki = 4149 nM T77913 C1JW2Q 13091358 Ki = 4149 nM T77913 CYN95Z 13091359 Ki = 977 nM T77913 CNW7P2 14248602 Ki = 25 nM T77913 CZQM08 14554127 Ki = 171 nM T77913 C8BF2P 15254720 Ki = 0.1585 nM T77913 CA5DC8 15542673 IC50 = 473 nM T77913 C4AD8Q 15542679 IC50 = 6.39 nM T77913 CZ0QW9 15542869 IC50 = 6.35 nM T77913 CL4J5G 15542871 IC50 = 6.89 nM T77913 CHDU67 15542874 IC50 = 6.67 nM T77913 CA09LW 15542879 IC50 = 285 nM T77913 CSM1B6 15542880 IC50 = 6.25 nM T77913 CGQU70 15542881 IC50 = 6.38 nM T77913 CO19UA 15595033 Ki = 2.4 nM T77913 CK6UH8 15749427 Ki = 11 nM T77913 C8IJ0O 15952316 Ki > 5000 nM T77913 CPR25X 15986917 Ki < 1995.26 nM T77913 CRBP36 15987008 Ki < 2511.89 nM T77913 C5KW3L 15987108 Ki < 2511.89 nM T77913 CXW37K 15987265 IC50 > 10000 nM T77913 CF6S2D 15987282 Ki < 1995.26 nM T77913 CXU15Z 15987451 Ki < 1995.26 nM T77913 C6V3WY 15987452 Ki = 1995.26 nM T77913 CG8KR9 16005860 IC50 = 6000 nM T77913 CH8K6G 16040671 Ki = 158.49 nM T77913 CT6AL1 16061961 Ki > 1000 nM T77913 CV36OS 16082828 IC50 = 6800 nM T77913 CHTO30 16082831 IC50 = 8500 nM T77913 CJ1DV9 16082833 EC50 > 10000 nM T77913 CD3E8L 16093484 Ki = 8 nM T77913 CS2HE1 16202149 Ki = 12.59 nM T77913 CZ2IS9 16660294 Ki > 10000 nM T77913 CY0UI3 16681693 Ki = 47 nM T77913 C08XJA 16718567 IC50 > 30000 nM T77913 CN3G6L 16722760 IC50 = 41 nM T77913 CDZC39 16722761 IC50 = 70 nM T77913 C7E6QC 17156312 Ki = 4570.88 nM T77913 CKH2W3 17178058 Ki = 316.23 nM T77913 CDA9E8 17590280 Ki = 537.03 nM T77913 C8QFZ1 17963141 Ki = 125.89 nM T77913 CP72GT 17963153 Ki = 15.85 nM T77913 C67NRA 17963183 Ki = 7.943 nM T77913 CHW4F9 17963196 Ki = 19.95 nM T77913 C8MJG3 17963199 Ki = 1000 nM T77913 C1H3UD 17963201 Ki = 19.95 nM T77913 CJS35W 17963208 Ki = 50.12 nM T77913 CBNK23 17963226 Ki = 25.12 nM T77913 C5ZT8C 17963227 Ki = 2.512 nM T77913 C9EVG1 17963258 Ki = 19.95 nM T77913 CQ7WR1 17963315 Ki = 31.62 nM T77913 C2V6WP 17963332 Ki = 19.95 nM T77913 COCE85 17963334 Ki = 50.12 nM T77913 C8KRN7 17963336 Ki = 19.95 nM T77913 CRYU86 17963347 Ki = 39.81 nM T77913 C2PWS7 17963363 Ki = 19.95 nM T77913 CO95VD 18333241 IC50 = 6.47 nM T77913 C20ZPL 18333379 IC50 = 6.6 nM T77913 CI2W9S 18337331 Ki = 1274 nM T77913 C9RWZ3 18382725 Ki = 1955 nM T77913 C6L3IF 18539962 Ki = 6025.6 nM T77913 CV0EI2 18672441 Ki = 5011.87 nM T77913 CJ6L5B 19426632 IC50 = 199.53 nM T77913 C6AOE8 19426635 IC50 = 10.72 nM T77913 CT1Q8M 19426644 IC50 = 3.02 nM T77913 CFYH89 19426650 IC50 > 1000 nM T77913 C9ODM1 19426658 IC50 > 1000 nM T77913 C7T8JC 19958494 Ki > 10000 nM T77913 C6LI5E 19958507 Ki > 10000 nM T77913 C74WSR 20659961 Ki = 441 nM T77913 C3T5HF 21509921 Ki = 50 nM T77913 CFN81Q 21527771 Ki = 698.6 nM T77913 CH59WN 21533446 Ki = 115 nM T77913 CT7XG9 21830793 Ki = 1030 nM T77913 CBN84K 22065997 Ki > 10000 nM T77913 C1R8KD 22322323 IC50 = 28 nM T77913 CL5D9B 22397436 Ki = 7.943 nM T77913 CDJ12S 22397445 Ki = 25.12 nM T77913 C81XUE 23027035 IC50 = 170 nM T77913 CR5H1I 23027211 IC50 = 390 nM T77913 CC2L1B 23027245 IC50 = 800 nM T77913 CG9M4Y 23027411 IC50 = 760 nM T77913 CC6R2O 23027527 IC50 = 810 nM T77913 CD14YL 23102733 Ki = 100 nM T77913 CU1T8V 23102749 Ki = 25.12 nM T77913 C3BP7D 23151209 IC50 > 10000 nM T77913 C2MJU1 23381046 Ki = 109 nM T77913 CL1YH7 23582308 Ki = 25.12 nM T77913 CZ1J7T 23722970 Ki = 6 nM T77913 CAD4S1 24740862 Ki = 826 nM T77913 C67YVI 24740863 Ki = 266 nM T77913 CRN13C 24748804 Ki = 1995.26 nM T77913 CTIF10 24748806 Ki < 3162.28 nM T77913 CMJU59 24748889 Ki < 1995.26 nM T77913 CB6R3K 24748890 Ki < 2511.89 nM T77913 C5EQ8T 24748892 Ki < 3162.28 nM T77913 CUMP36 24748894 Ki < 2511.89 nM T77913 C1XN4V 24748896 Ki < 2511.89 nM T77913 CFR1S3 24748988 Ki < 2511.89 nM T77913 CG43ZS 24748989 Ki < 2511.89 nM T77913 C96KDH 24748992 Ki < 1995.26 nM T77913 CH8N1W 24748993 Ki < 2511.89 nM T77913 CQF29T 24749076 Ki < 1995.26 nM T77913 CU0GX7 24749078 Ki < 1995.26 nM T77913 CGD2I7 24749080 Ki < 1995.26 nM T77913 CB8DF0 24749082 Ki < 3162.28 nM T77913 C9XS6U 24749083 Ki < 2511.89 nM T77913 CKVA89 24749182 Ki < 2511.89 nM T77913 CRGJ52 24749183 Ki < 2511.89 nM T77913 C13GRZ 24749184 Ki < 1995.26 nM T77913 C8ZE6H 24749185 Ki = 2511.89 nM T77913 CG9I8K 24749186 Ki < 2511.89 nM T77913 CF8W2P 24749291 Ki < 2511.89 nM T77913 CTB38H 24749292 Ki < 2511.89 nM T77913 CET71X 24749293 Ki < 2511.89 nM T77913 CAE9S7 24749294 Ki < 2511.89 nM T77913 CKV83Y 24749295 Ki < 2511.89 nM T77913 C6S0OJ 24749401 Ki < 2511.89 nM T77913 CSG9V8 24749508 Ki = 1995.26 nM T77913 CWTB59 24749606 Ki = 1258.93 nM T77913 CLFS68 24749607 Ki = 1995.26 nM T77913 CHYC87 24749609 Ki = 1995.26 nM T77913 CY53AF 24749610 Ki < 2511.89 nM T77913 CT93NP 24749721 Ki < 1995.26 nM T77913 C7EGL2 24749724 Ki < 2511.89 nM T77913 CW19JN 24749726 Ki < 2511.89 nM T77913 CI6W7D 24749841 Ki < 2511.89 nM T77913 CV20EP 24749844 Ki < 1995.26 nM T77913 CYI79E 24749958 Ki < 3162.28 nM T77913 CGT53R 24749959 Ki < 2511.89 nM T77913 C20QND 24749960 Ki < 1995.26 nM T77913 CSXA65 24749962 Ki < 1584.89 nM T77913 CNOX23 24750086 Ki < 1584.89 nM T77913 C1XRY9 24750087 Ki < 2511.89 nM T77913 C89WKU 24750088 Ki < 2511.89 nM T77913 C0I2HU 24769156 Ki = 110 nM T77913 CUX7C3 24803316 Ki = 39.81 nM T77913 C1QTN4 24803480 Ki = 39.81 nM T77913 CTU67D 24803482 Ki = 25.12 nM T77913 C31QHW 24803483 Ki = 12.59 nM T77913 C3RYC2 24803638 Ki = 7.943 nM T77913 CI4EA6 24803639 Ki = 12.59 nM T77913 CJ07ES 24803641 Ki = 50.12 nM T77913 C04KHJ 24803797 Ki = 15.85 nM T77913 CY26TH 24803798 Ki = 15.85 nM T77913 C50BOH 24803799 Ki = 19.95 nM T77913 C2AKX9 24804150 Ki = 17.38 nM T77913 CDC91N 24839550 Ki = 125.89 nM T77913 CY21RE 24841480 Ki = 29 nM T77913 C3C0KP 24894134 EC50 > 50000 nM T77913 CZPW63 24936097 Ki > 1000 nM T77913 CQ52SD 24936098 Ki > 1000 nM T77913 CA20NZ 25025581 Ki = 1000 nM T77913 C2G1JK 25053351 Ki > 10000 nM T77913 C51OJR 25099115 IC50 > 10000 nM T77913 C7NJ1B 25109291 Ki = 3548.13 nM T77913 CML6G5 25128822 Ki = 9120.11 nM T77913 C6HD3B 25147771 Ki = 97.72 nM T77913 C1RU5I 25147772 Ki = 19.95 nM T77913 C5C7GH 25184832 Ki = 50.12 nM T77913 C78HME 25212275 Ki = 390 nM T77913 CE6Z9I 25212276 Ki = 40 nM T77913 CJ1Z9H 25216680 Ki = 7230 nM T77913 C1T3LR 25218143 Ki = 9620 nM T77913 CPI03N 25218397 Ki > 10000 nM T77913 CL1R3Q 25218401 Ki = 8750 nM T77913 C2QLS7 25375331 Ki > 10000 nM T77913 CRB9W7 25450664 Ki = 2758 nM T77913 C8FWE5 25456694 Ki > 10000 nM T77913 CEK31Q 25487292 Ki > 10000 nM T77913 CN39GC 25491778 Ki = 3265 nM T77913 CAQ5S0 26191740 Ki = 10000 nM T77913 C1QT2Y 28071610 Ki > 10000 nM T77913 CU9PY2 28357663 Ki = 280 nM T77913 CYKH58 28390601 Ki = 125 nM T77913 C73KWR 29136870 Ki = 61.66 nM T77913 C9MZ5R 29983056 Ki > 10000 nM T77913 CEZ1A6 32718395 Ki > 10000 nM T77913 CW04EV 40011786 Ki = 3235.94 nM T77913 C8G7QX 42625303 EC50 = 3467.37 nM T77913 C75WJN 42625304 EC50 = 2570.4 nM T77913 C0BW6J 42625384 EC50 = 12882.5 nM T77913 CID4J1 42625386 EC50 = 2187.76 nM T77913 C4W5PM 42626110 EC50 = 1698.24 nM T77913 CY7W2J 42631003 IC50 = 146 nM T77913 C0AI7N 43229249 Ki = 63.1 nM T77913 CJ41QV 44126269 IC50 = 112 nM T77913 CG1VP5 44126270 IC50 = 104 nM T77913 CN3IA4 44126272 IC50 = 68 nM T77913 CY6PC2 44126325 IC50 = 66 nM T77913 C32MRX 44126326 IC50 = 30 nM T77913 CQ28AG 44126327 IC50 = 98 nM T77913 CNF19Z 44126328 IC50 = 31 nM T77913 CHFE79 44126329 IC50 = 500 nM T77913 C2Q0UX 44126330 IC50 = 500 nM T77913 C7I9YB 44189144 IC50 = 40 nM T77913 CVG6X1 44209472 Ki = 262 nM T77913 CD5AB7 44209480 Ki = 167 nM T77913 CPI9X4 44224259 IC50 = 100 nM T77913 CH59RP 44247803 Ki = 0.6 nM T77913 C7MY2N 44247806 Ki = 1.3 nM T77913 CF9TE1 44247935 Ki = 0.9 nM T77913 C85DHY 44250284 Ki = 3.9 nM T77913 C8P2LE 44250288 IC50 > 10000 nM T77913 CEL7B6 44275464 Ki < 1905.46 nM T77913 CE20CZ 44275807 Ki = 2344.23 nM T77913 CC2OD4 44278111 Ki > 10000 nM T77913 CRMA84 44278114 Ki > 10000 nM T77913 CF0Y4M 44278115 Ki > 10000 nM T77913 CZ5P6U 44288769 Ki = 302 nM T77913 CZ7O4D 44288847 Ki = 91 nM T77913 C6DYQ1 44288874 Ki = 108 nM T77913 CAG7E1 44288877 Ki = 616 nM T77913 CQ74LV 44288917 Ki = 63 nM T77913 CQ3Y5R 44288945 Ki = 19 nM T77913 C5ZL4A 44289035 Ki = 355 nM T77913 CA0DN5 44304003 Ki = 45708.82 nM T77913 C3Z5DG 44304012 Ki = 35481.34 nM T77913 CZ5X0G 44304013 Ki = 21877.62 nM T77913 CK63QN 44304014 Ki = 16218.1 nM T77913 C1P7BD 44304021 Ki = 354.81 nM T77913 CNKS56 44304030 Ki = 12022.64 nM T77913 CJF2S5 44304031 Ki = 616.6 nM T77913 CK7Q8R 44304032 Ki = 4265.8 nM T77913 CGA15P 44304035 Ki = 933.25 nM T77913 CY2JQ9 44304036 Ki = 977.24 nM T77913 CGP5R0 44304037 Ki = 741.31 nM T77913 C6D4QK 44304049 Ki = 4570.88 nM T77913 C95EPL 44304056 Ki = 46773.51 nM T77913 C8FUS4 44304064 Ki = 9772.37 nM T77913 CTZB24 44304066 Ki = 13489.63 nM T77913 C1I2VN 44304067 Ki = 100000 nM T77913 C7BOY8 44304068 Ki = 14454.4 nM T77913 CS7V9L 44304079 Ki = 933.25 nM T77913 CCH2E6 44304088 Ki = 602.56 nM T77913 C9IM6V 44304090 Ki = 1412.54 nM T77913 CY0SG5 44304091 Ki = 501.19 nM T77913 CP3DB1 44304211 Ki = 2089.3 nM T77913 CL9F2Z 44304223 Ki = 457.09 nM T77913 CP0Z1H 44304243 Ki = 660.69 nM T77913 CU6LJ1 44304244 Ki = 2238.72 nM T77913 CQ86HY 44304245 Ki = 56.23 nM T77913 CY5NQ8 44304246 Ki = 104.71 nM T77913 CKE47A 44304247 Ki = 398.11 nM T77913 CG5TJ8 44304256 Ki = 3388.44 nM T77913 C1GQH4 44304259 Ki = 79.43 nM T77913 C4RL7Y 44304269 Ki = 478.63 nM T77913 CLH2M5 44304270 Ki = 97.72 nM T77913 C2RPN4 44304277 Ki = 34673.69 nM T77913 CVXS65 44304282 Ki = 380.19 nM T77913 C0A8SI 44304283 Ki = 562.34 nM T77913 C6G3YS 44304284 Ki = 812.83 nM T77913 CQU2W4 44304287 Ki = 74.13 nM T77913 CYX69C 44304288 Ki = 1778.28 nM T77913 CUN8B6 44304291 Ki = 3981.07 nM T77913 CK5OM8 44304293 Ki = 4365.16 nM T77913 C9U0HX 44304294 Ki = 1995.26 nM T77913 CC76QK 44304295 Ki = 10000 nM T77913 CSR0G4 44304303 Ki = 10000 nM T77913 CBH73L 44304304 Ki = 426.58 nM T77913 C97BJW 44304307 Ki = 870.96 nM T77913 CHR62F 44304308 Ki = 1023.29 nM T77913 CUWM24 44304309 Ki = 208.93 nM T77913 C1J2NZ 44304310 Ki = 1047.13 nM T77913 CFSR60 44304311 Ki = 100000 nM T77913 C13YKA 44304312 Ki = 9332.54 nM T77913 CJ0DI3 44304313 Ki = 9772.37 nM T77913 CZ1RI6 44304316 Ki = 46773.51 nM T77913 C5W1TM 44304318 Ki = 1513.56 nM T77913 CJY49E 44304319 Ki = 1737.8 nM T77913 C3YC4E 44304320 Ki = 4677.35 nM T77913 C7RJ8O 44304325 Ki = 1584.89 nM T77913 CVT19R 44304327 Ki = 5495.41 nM T77913 CBJK06 44304329 Ki = 37153.52 nM T77913 C3B0GW 44304331 Ki = 10000 nM T77913 C3-FEB-02 44304332 Ki = 95499.26 nM T77913 C6J5OZ 44304348 Ki = 46773.51 nM T77913 CN2W8Q 44304349 Ki = 9332.54 nM T77913 CC9PT2 44304357 Ki = 10232.93 nM T77913 CSX2L0 44304376 Ki = 416.87 nM T77913 CEWD86 44304377 Ki = 2041.74 nM T77913 CZ86DV 44304378 Ki = 724.44 nM T77913 C0TYR3 44304382 Ki = 1202.26 nM T77913 CH23XB 44304383 Ki = 275.42 nM T77913 CP7I3Z 44304385 Ki = 309.03 nM T77913 C7ZF0Q 44304387 Ki = 2238.72 nM T77913 CV3O9C 44304393 Ki = 21379.62 nM T77913 CZ0Q7N 44304399 Ki = 575.44 nM T77913 CEQO51 44304402 Ki = 60.26 nM T77913 CT7L5H 44304412 Ki = 3311.31 nM T77913 C1KIA2 44304415 Ki = 16982.44 nM T77913 COP9L3 44304431 Ki = 16982.44 nM T77913 CS20NC 44304437 Ki = 21379.62 nM T77913 CV7U0X 44304438 Ki = 1096.48 nM T77913 C9OES6 44304439 Ki = 56.23 nM T77913 C4KX8A 44304445 Ki = 8128.31 nM T77913 CKY4V8 44304449 Ki = 4677.35 nM T77913 CF2X5I 44304450 Ki = 19054.61 nM T77913 C95OLE 44304451 Ki = 16595.87 nM T77913 C5I2QL 44304457 Ki = 1071.52 nM T77913 CB6G5H 44304459 Ki = 562.34 nM T77913 C6JT1P 44304462 Ki = 46773.51 nM T77913 CUR3O7 44304475 Ki = 1659.59 nM T77913 C19UMQ 44304494 Ki = 6760.83 nM T77913 CQ6A4T 44304516 Ki = 21877.62 nM T77913 CMGY49 44304558 Ki = 1905.46 nM T77913 CX97UN 44304560 Ki = 12589.25 nM T77913 CO6ZF2 44304719 Ki = 95499.26 nM T77913 CR2YO1 44304741 Ki = 2290.87 nM T77913 C57WXT 44304743 Ki = 9772.37 nM T77913 CN51UA 44304751 Ki = 288.4 nM T77913 CP05OY 44304752 Ki = 8128.31 nM T77913 CNEK74 44304753 Ki = 3311.31 nM T77913 CE6P5V 44304760 Ki = 14454.4 nM T77913 C6WM1H 44304978 Ki = 26302.68 nM T77913 C5OYK1 44304990 Ki = 13489.63 nM T77913 CDHT79 44304991 Ki = 11220.18 nM T77913 CT63YZ 44307779 Ki = 15733 nM T77913 CENZ76 44312371 Ki = 190 nM T77913 CAJL61 44312568 Ki = 660 nM T77913 C04AFJ 44312705 Ki = 4 nM T77913 C5MOH0 44312748 Ki = 180 nM T77913 CK5WM1 44313266 Ki = 189 nM T77913 C1L3DB 44318442 IC50 > 1000 nM T77913 CV8WZ0 44318454 IC50 = 2.57 nM T77913 CMQW13 44318461 IC50 = 6.026 nM T77913 CPIT23 44318554 IC50 = 1.738 nM T77913 C75CNK 44318581 IC50 = 1.288 nM T77913 C84MTV 44318695 IC50 = 7.943 nM T77913 C8LK5W 44318820 IC50 = 15.85 nM T77913 C35OHA 44318834 IC50 = 15.49 nM T77913 CWN39R 44318841 IC50 = 11.75 nM T77913 CXJL56 44318842 IC50 = 5.888 nM T77913 C7CTF9 44318853 IC50 > 1000 nM T77913 CM39LE 44319098 IC50 = 37.15 nM T77913 C5NG8E 44319099 IC50 > 1000 nM T77913 C3RV7M 44319119 IC50 = 14.45 nM T77913 CY8L5E 44319120 IC50 = 2.291 nM T77913 CE0I4R 44319133 IC50 = 3.802 nM T77913 C9MY2X 44319134 IC50 = 47.86 nM T77913 CW16JD 44324737 Ki = 460 nM T77913 CA84SN 44324765 Ki > 1000 nM T77913 COA3H4 44324800 Ki = 113 nM T77913 CY04JW 44324972 Ki > 1000 nM T77913 C29NRF 44326124 Ki = 47.1 nM T77913 CHR3P2 44326125 Ki = 1.9 nM T77913 C0C1LX 44326219 Ki = 471 nM T77913 CTC70Y 44326298 Ki = 27 nM T77913 C2OZT8 44326319 Ki = 0.7 nM T77913 C8TQL9 44326320 Ki = 32.6 nM T77913 C0GJ3W 44326321 Ki = 14 nM T77913 CUJ74H 44326336 Ki = 4.3 nM T77913 CGE89D 44326357 Ki = 6 nM T77913 C3VT2B 44326358 Ki = 9.6 nM T77913 C3A1WX 44326390 Ki = 2.36 nM T77913 C9KA7Y 44326405 Ki = 20.6 nM T77913 CCSV14 44326407 Ki = 3.7 nM T77913 CY4C9X 44326422 Ki = 9.3 nM T77913 CTGR29 44326427 Ki = 3 nM T77913 CKHM97 44326433 Ki = 29.7 nM T77913 CIC4V1 44326442 Ki = 1.2 nM T77913 CW2A8X 44326690 Ki = 3.74 nM T77913 C5HW0O 44326705 Ki = 0.63 nM T77913 CC6BR5 44327909 IC50 = 446 nM T77913 CKW8A5 44328177 IC50 = 158 nM T77913 CI0TC6 44328187 IC50 = 7.33 nM T77913 C69TAU 44328188 IC50 = 6.2 nM T77913 CS13PB 44328320 IC50 = 6 nM T77913 CX6BT1 44328321 IC50 = 5.04 nM T77913 CG6Z4H 44333987 Ki = 60000 nM T77913 CA7OE5 44333988 Ki = 7400 nM T77913 CGR23Y 44334025 Ki = 4500 nM T77913 C46JFI 44334035 Ki = 37000 nM T77913 C9MFY5 44334036 Ki = 13000 nM T77913 CZ9LJ8 44334037 Ki = 11000 nM T77913 C37JOG 44334038 Ki = 8900 nM T77913 C2L8JG 44334042 Ki = 6200 nM T77913 CJ96XL 44334212 Ki = 2300 nM T77913 CGPL96 44334214 Ki = 14000 nM T77913 CJB65X 44334234 Ki = 91000 nM T77913 C13TRB 44334235 Ki = 16000 nM T77913 C9PY0X 44334252 Ki = 80000 nM T77913 CY8XM2 44334265 Ki = 10000 nM T77913 CP4W5X 44334281 Ki = 56000 nM T77913 C9BS4V 44334368 Ki = 1500 nM T77913 CM57UH 44334369 Ki = 2300 nM T77913 C9M1NZ 44334395 Ki = 9200 nM T77913 C1EQY2 44334396 Ki = 9400 nM T77913 CC1RW3 44334406 Ki = 2500 nM T77913 C18SHG 44334407 Ki = 3600 nM T77913 CDQ72F 44334430 Ki = 9100 nM T77913 CS7YO0 44334503 Ki = 43000 nM T77913 CM15VJ 44334521 Ki = 90000 nM T77913 CFHU75 44334556 Ki = 75000 nM T77913 C9XC5R 44334781 Ki = 4400 nM T77913 CXD0C7 44334782 Ki = 5500 nM T77913 C1L3GT 44335172 Ki = 758.58 nM T77913 C6KCD9 44335185 Ki = 181.97 nM T77913 C24HSP 44335222 Ki = 3715.35 nM T77913 C4BLC5 44335225 Ki = 2884.03 nM T77913 C8HYU5 44335237 Ki = 27.54 nM T77913 C1TL7P 44335238 Ki = 3981.07 nM T77913 C51LMP 44335336 Ki = 3548.13 nM T77913 C7R2BK 44335350 Ki = 354.81 nM T77913 CDFA49 44335351 Ki = 354.81 nM T77913 CCY4I9 44335368 Ki = 380.19 nM T77913 CCI26P 44335384 Ki = 3467.37 nM T77913 CNF4S6 44335387 Ki = 158.49 nM T77913 CO75LT 44335389 Ki = 162.18 nM T77913 C2ZN6D 44335405 Ki = 8912.51 nM T77913 C18ONA 44335407 Ki = 436.52 nM T77913 C7LH1C 44335412 Ki = 81.28 nM T77913 C89TNO 44335428 Ki = 1479.11 nM T77913 CPQW41 44335430 Ki = 446.68 nM T77913 C04MTD 44335456 Ki = 575.44 nM T77913 CO0GR9 44335463 Ki = 501.19 nM T77913 CMD1U0 44335483 Ki = 7762.47 nM T77913 C12MNS 44335558 Ki = 426.58 nM T77913 CJX50C 44335559 Ki = 275.42 nM T77913 CN9JI6 44335571 Ki = 3235.94 nM T77913 C6N3XK 44345317 IC50 = 16.6 nM T77913 CCU89V 44350664 Ki = 973.5 nM T77913 C8WV2Q 44369359 IC50 = 50118.72 nM T77913 CU67KP 44389292 Ki = 9.55 nM T77913 CU2X6H 44389293 Ki = 5.01 nM T77913 CF27BX 44389301 Ki = 7.59 nM T77913 CTG4C7 44389302 Ki = 17.8 nM T77913 CXT7P9 44395497 Ki = 30 nM T77913 C3QW5V 44395530 Ki = 9 nM T77913 C3RV6T 44395741 Ki = 157.6 nM T77913 CX7O9S 44401041 Ki = 7.5 nM T77913 C5XC2B 44401042 Ki = 14 nM T77913 CD56EA 44401105 Ki = 42 nM T77913 CW3PC2 44401106 Ki = 1.2 nM T77913 C9WH7P 44401164 Ki = 0.52 nM T77913 C9CWX1 44401194 Ki = 33 nM T77913 CXT84G 44401243 Ki = 4.3 nM T77913 C1B4QL 44403095 Ki > 10000 nM T77913 C1YL7Z 44403098 Ki > 10000 nM T77913 CFV98A 44403101 Ki > 10000 nM T77913 C6OY9S 44403102 Ki > 10000 nM T77913 CH4SX6 44403105 Ki > 10000 nM T77913 C12FIH 44403106 Ki > 10000 nM T77913 C4LKC1 44404394 Ki > 10000 nM T77913 C3EJ4G 44404396 Ki > 10000 nM T77913 CSH9J2 44404954 Ki = 20 nM T77913 C3VE2D 44449768 Ki = 10 nM T77913 C83ICG 44449794 Ki = 26 nM T77913 C52HPA 44450154 Ki = 10 nM T77913 CAW6S7 44450181 Ki = 10 nM T77913 C4M0PG 44450184 Ki = 10 nM T77913 CSQR06 44450212 Ki = 10 nM T77913 CB1MX2 44454118 Ki > 5011.87 nM T77913 CR3IC6 44454120 Ki = 2511.89 nM T77913 C5B0IF 44454150 Ki < 1584.89 nM T77913 CRD82N 44454166 Ki > 2511.89 nM T77913 CMVS90 44454167 Ki > 3162.28 nM T77913 CW4S3P 44454190 Ki = 794.33 nM T77913 C7H3CL 44454192 Ki > 2511.89 nM T77913 CU0N1E 44454217 Ki > 2511.89 nM T77913 C9DBA3 44454218 Ki > 2511.89 nM T77913 CK01QH 44454219 Ki > 2511.89 nM T77913 CLO6X0 44454223 Ki = 1000 nM T77913 CECR53 44454247 Ki > 2511.89 nM T77913 CD4ZU7 44454248 Ki > 2511.89 nM T77913 CS2N1D 44454275 Ki > 1584.89 nM T77913 CJ5XB1 44454278 Ki = 1995.26 nM T77913 C4GON0 44454309 Ki = 158.49 nM T77913 C91PHS 44454318 Ki < 3162.28 nM T77913 CT50UC 44454320 Ki < 3162.28 nM T77913 C35WYK 44454339 Ki > 2511.89 nM T77913 CZO96M 44454340 Ki > 2511.89 nM T77913 C2CIO7 44454351 Ki = 794.33 nM T77913 C9AH1O 44454352 Ki < 3162.28 nM T77913 CM8H2G 44454353 Ki = 1995.26 nM T77913 C1EZP7 44454358 Ki < 3162.28 nM T77913 CEB84V 44454371 Ki > 3981.07 nM T77913 C5EV7Z 44454381 Ki < 3162.28 nM T77913 CWC92Y 44454382 Ki = 1000 nM T77913 CH0S2F 44454384 Ki < 3162.28 nM T77913 C32LHE 44454400 Ki > 2511.89 nM T77913 CG18KC 44454401 Ki = 1584.89 nM T77913 CI0CJ9 44454402 Ki > 2511.89 nM T77913 CP34QH 44454403 Ki > 3162.28 nM T77913 CW4OX5 44454418 Ki < 2511.89 nM T77913 CW1I4Z 44454420 Ki < 2511.89 nM T77913 C8TJW4 44454434 Ki = 3162.28 nM T77913 CX9U8I 44454443 Ki = 2511.89 nM T77913 CXA7W2 44454458 Ki = 1000 nM T77913 CBGJ08 44454459 Ki > 501.19 nM T77913 CZL97F 44455426 Ki = 374 nM T77913 C12XGE 44456400 Ki > 10000 nM T77913 C5RO6E 44461290 IC50 > 1000 nM T77913 CC9JB4 44461357 IC50 = 102.33 nM T77913 CI85BO 44461456 IC50 = 61.66 nM T77913 CE12QP 44461565 IC50 = 676.08 nM T77913 CQ2IX7 44461606 IC50 = 83.18 nM T77913 C5RM2Q 44461613 IC50 = 151.36 nM T77913 CJ91XI 44461619 IC50 > 1000 nM T77913 CQX62Y 44461622 IC50 = 13.49 nM T77913 C80PVC 44461625 IC50 > 1000 nM T77913 CT09SU 44461626 IC50 > 1000 nM T77913 CR54MO 44461647 IC50 > 1000 nM T77913 C5P3AW 44461799 IC50 > 1000 nM T77913 C52INO 44461800 IC50 = 26.3 nM T77913 CQ0WM7 44469273 IC50 > 5000 nM T77913 C4DL5C 44469677 IC50 > 10000 nM T77913 CK10AW 44478385 Ki = 25703.96 nM T77913 CM23CO 44521013 Ki = 6 nM T77913 CVA67X 44568347 Ki = 430 nM T77913 CRCH48 44582675 Ki = 509 nM T77913 CEJ4R8 44582676 Ki = 944 nM T77913 C5QB4K 44582678 Ki = 439 nM T77913 C01RCI 44582705 Ki = 665 nM T77913 CP6ZA9 44591012 Ki = 559 nM T77913 CU37BO 44591098 Ki = 686 nM T77913 CU48CL 44591099 Ki = 79 nM T77913 C7H9SE 44591134 Ki = 205 nM T77913 C6RLW0 44591135 Ki = 295 nM T77913 C7NH9W 44622869 Ki = 16 nM T77913 C8B0HO 44622872 Ki = 39 nM T77913 CR3PL6 44665680 Ki < 1000 nM T77913 CYXD79 45257131 Ki > 1000 nM T77913 C07WHQ 45257132 Ki > 1000 nM T77913 CY25IH 45257133 Ki > 1000 nM T77913 C08WYZ 45267326 IC50 = 23 nM T77913 CEJ8T4 45267329 IC50 = 69 nM T77913 C6SV5O 45267774 Ki = 75.2 nM T77913 CHQ05B 45267775 IC50 = 80.5 nM T77913 C6W9OC 45268181 IC50 = 23 nM T77913 C9V0LE 45268182 IC50 > 500 nM T77913 CGNJ76 45268185 IC50 = 105 nM T77913 C6KAT3 45268186 IC50 = 41 nM T77913 C9B5EH 45268653 Ki = 3.2 nM T77913 C65LBY 45268662 Ki = 2.4 nM T77913 CBC26P 45269062 IC50 = 46 nM T77913 CNJ79X 45269063 IC50 = 53 nM T77913 C8I4DX 45269069 IC50 > 500 nM T77913 C3AF9J 45269070 IC50 = 124 nM T77913 C21OMZ 45269073 IC50 = 123 nM T77913 CCFG82 45269436 IC50 = 3.3 nM T77913 CU8HZ3 45269933 IC50 = 41 nM T77913 C8GQ7J 45270330 Ki = 14.1 nM T77913 C48BMQ 45270339 Ki = 6.6 nM T77913 CFZ01K 45270350 IC50 = 4.4 nM T77913 C6WP0Z 45270750 IC50 = 37 nM T77913 C8CGE1 45270753 IC50 = 35 nM T77913 C4QEG5 45270755 IC50 = 72 nM T77913 C18WQE 45271166 Ki = 7.1 nM T77913 CW6HL5 45271167 Ki = 3.6 nM T77913 CU9C4I 45272046 Ki = 2.2 nM T77913 CAY8I7 45272070 Ki = 18.3 nM T77913 CO4F0Z 45272487 IC50 = 323 nM T77913 C62IGT 45272875 Ki = 1.8 nM T77913 C3GUK4 45272876 Ki = 1.5 nM T77913 CBE0M8 45272877 Ki = 2.4 nM T77913 CR04WH 45272878 Ki = 14.1 nM T77913 CZ7N8Q 45272889 Ki = 4.5 nM T77913 CK2B5U 45272890 Ki = 2.9 nM T77913 C8TC4R 45272894 Ki = 1.3 nM T77913 CA0SD1 45272895 Ki = 6.9 nM T77913 CPF5S7 45273362 IC50 = 88 nM T77913 C0U6LA 45273370 IC50 > 1000 nM T77913 C5E2XR 45273828 Ki = 59.3 nM T77913 CE71LQ 45273833 Ki = 2.8 nM T77913 CMNA70 45358442 Ki = 2.512 nM T77913 CGLF37 45484995 IC50 = 920 nM T77913 CGOS24 45485061 IC50 = 1210 nM T77913 CLX9C8 45485062 IC50 = 1600 nM T77913 C3AT2W 45485462 Ki = 61 nM T77913 CIG91B 45485473 Ki = 20 nM T77913 CFN4G6 45485525 Ki = 121 nM T77913 CR9V5P 45485529 Ki = 64 nM T77913 CCB1R8 45485535 Ki = 155 nM T77913 C3QU2C 45487384 IC50 > 5000 nM T77913 CXT96Y 45815848 Ki = 1191 nM T77913 CV7C2M 45827434 Ki > 10000 nM T77913 C0FE4R 45833388 Ki = 707.95 nM T77913 C2L5UH 46182745 IC50 = 8150 nM T77913 C16KNO 46216770 Ki = 242 nM T77913 CRT07W 46216771 Ki = 725 nM T77913 C7M9XU 46216789 Ki = 964 nM T77913 CZJH90 46224877 IC50 = 33 nM T77913 CFL32X 46224878 IC50 = 345 nM T77913 C5FQ4S 46224879 IC50 = 154 nM T77913 CAZX21 46225000 IC50 = 131 nM T77913 CDBP61 46225002 IC50 = 35 nM T77913 C38OVM 46225027 IC50 = 32 nM T77913 CTE69Y 46230651 Ki = 2640 nM T77913 CU15OL 46235428 EC50 > 10000 nM T77913 CN75IJ 46830167 EC50 = 831.76 nM T77913 CC68WI 46830289 Ki = 4.4 nM T77913 CP6DN0 46861858 Ki = 0.8 nM T77913 CW1FS9 46861860 Ki = 0.5 nM T77913 C2QH7O 46865650 Ki = 1 nM T77913 CC5KR7 46865978 Ki = 2.5 nM T77913 C2MC4K 46881463 Ki = 1995.26 nM T77913 CSQ4C9 46881468 Ki = 2511.89 nM T77913 C6KBJ2 46882133 Ki = 923 nM T77913 CNL16U 46882180 Ki = 1374 nM T77913 CCX75M 46882181 Ki = 199 nM T77913 C2BOJ6 46882182 Ki = 5000 nM T77913 C9ASC1 46882224 Ki = 38400 nM T77913 CD0VH7 46882664 Ki = 1013 nM T77913 CW6A9I 46884062 Ki = 32000 nM T77913 C04JMO 46884063 Ki = 3.9 nM T77913 CR1Z8E 46884119 Ki = 38 nM T77913 CR0CQ9 46884120 Ki = 5 nM T77913 C9OYT5 46884152 Ki = 2.7 nM T77913 CCI32B 46884153 Ki = 8 nM T77913 C2JQE7 46884154 Ki = 120 nM T77913 C20HET 46884155 Ki = 17 nM T77913 C0HYN3 46884200 Ki = 2.9 nM T77913 CM6A8S 46884201 Ki = 4.6 nM T77913 CW94IK 46884202 Ki = 5.2 nM T77913 C3QT0U 46884239 Ki = 122 nM T77913 COPQ16 46884600 Ki = 12 nM T77913 C85MOA 46884637 Ki = 63 nM T77913 C36NKV 46884638 Ki = 35 nM T77913 CQ84IF 46884639 Ki = 2.2 nM T77913 CZGS15 46884640 Ki = 7.7 nM T77913 CZ72SW 46884641 Ki = 15 nM T77913 CA3Z6G 46884666 Ki = 0.8 nM T77913 C8DBY0 46884667 Ki = 3.1 nM T77913 CU3BG6 46884668 Ki = 11.9 nM T77913 CPG14Q 46884669 Ki = 8.9 nM T77913 C7R9AK 46884670 Ki = 1.4 nM T77913 C64KNW 46884698 Ki = 1.5 nM T77913 C0ASK4 46884699 Ki = 4.2 nM T77913 CYNU85 46884731 Ki = 3.1 nM T77913 CJ6O8D 46884732 Ki = 2.7 nM T77913 C9QT7G 46884733 Ki = 1.3 nM T77913 CL6Z7Q 46884734 Ki = 0.7 nM T77913 C6PRX8 46884735 Ki = 0.3 nM T77913 CWK8I4 46884736 Ki = 2.2 nM T77913 CB29TI 46887041 EC50 = 6165.95 nM T77913 C9P3CV 46887042 EC50 = 89.13 nM T77913 C12SYH 46887043 EC50 = 66.07 nM T77913 CQJ8W2 46887076 EC50 > 10000 nM T77913 CAG89L 46887077 EC50 > 10000 nM T77913 COK81L 46887078 EC50 > 10000 nM T77913 CB09SD 46887079 EC50 > 10000 nM T77913 CK0S2U 46887080 EC50 > 10000 nM T77913 CLPJ52 46887115 EC50 > 10000 nM T77913 CJK1Z5 46888857 Ki = 0.9 nM T77913 CX92WH 46889257 Ki = 8.4 nM T77913 C01DMO 46889258 Ki = 4.8 nM T77913 COR71G 46890166 EC50 > 10000 nM T77913 C8FR9E 46890592 EC50 > 10000 nM T77913 CDV30W 46912441 Ki > 1000 nM T77913 CAQ0E9 46912442 Ki > 1000 nM T77913 C6F2MP 46929551 Ki > 10000 nM T77913 CT3UX6 46929553 Ki > 10000 nM T77913 CZJ2G8 46929554 Ki = 540 nM T77913 C40EGB 46929647 Ki = 280 nM T77913 CB95RA 46929648 Ki = 48 nM T77913 CG7WR2 46933089 Ki = 25.12 nM T77913 CW4N5K 46933090 Ki = 39.81 nM T77913 CZO5F8 46933091 Ki = 79.43 nM T77913 C6SJ7N 46967967 Ki = 1778.28 nM T77913 C3XFG4 47029237 Ki > 10000 nM T77913 CPFY62 49782791 Ki = 3.6 nM T77913 CKGU71 49782792 Ki = 2.5 nM T77913 CNE84I 49782794 Ki = 4.5 nM T77913 CS09QO 49782998 Ki = 5 nM T77913 CD53RT 49833882 Ki = 63.1 nM T77913 C5Y4DE 49833883 Ki = 39.81 nM T77913 CGT73Y 49833884 Ki = 50.12 nM T77913 CKL16R 49833886 Ki = 125.89 nM T77913 C3KSZ8 49834050 Ki = 50.12 nM T77913 C9QS2K 49834051 Ki = 12.59 nM T77913 CF4SX0 49834052 Ki = 31.62 nM T77913 C52GPW 49834053 Ki = 39.81 nM T77913 CO20JE 49836187 Ki = 25.12 nM T77913 CG0LF8 49836189 Ki = 158.49 nM T77913 C0UI3V 49836294 Ki = 15.85 nM T77913 CT7CV0 49836295 Ki = 19.95 nM T77913 CVG9X5 49836296 Ki = 39.81 nM T77913 C5E2ZK 49836298 Ki = 39.81 nM T77913 CYJW87 49836299 Ki = 50.12 nM T77913 C0MS8L 49836300 Ki = 50.12 nM T77913 CKS86Q 49836409 Ki = 50.12 nM T77913 C8E6WA 49836410 Ki = 39.81 nM T77913 CE0PN6 49836411 Ki = 25.12 nM T77913 C0I4EC 49836412 Ki = 19.95 nM T77913 C5HU1D 49836413 Ki = 794.33 nM T77913 C1UGC7 49836414 Ki = 63.1 nM T77913 C5ZV2Y 49836522 Ki = 100 nM T77913 C1JTH9 49836524 Ki = 15.85 nM T77913 C90XTY 49836525 Ki = 12.59 nM T77913 CK5QW9 49836526 Ki = 31.62 nM T77913 C8RL7C 49836527 Ki = 39.81 nM T77913 CNM9X8 49836528 Ki = 31.62 nM T77913 COK75S 49836633 Ki = 6.31 nM T77913 CZ6F7L 49836634 Ki = 316.23 nM T77913 CRM28S 49836635 Ki = 199.53 nM T77913 CA6QB8 49836636 Ki = 100 nM T77913 CB81YG 49836637 Ki = 50.12 nM T77913 CX43UC 49836639 Ki = 79.43 nM T77913 CEBP01 49836737 Ki = 158.49 nM T77913 CCMJ40 49836738 Ki = 125.89 nM T77913 CY1UR9 49836739 Ki = 79.43 nM T77913 C3OK9Y 49836740 Ki = 1000 nM T77913 C26NFU 49836741 Ki = 199.53 nM T77913 C6YM8W 49836842 Ki = 199.53 nM T77913 CG97QN 49841719 Ki = 7373 nM T77913 CZ3T1W 49841845 Ki = 6422 nM T77913 C3SBE0 49841846 Ki = 2800 nM T77913 CZ2SA8 49864841 Ki = 0.631 nM T77913 C2OCZ3 49864885 Ki = 50.12 nM T77913 CS4Z8A 49864886 Ki = 19.95 nM T77913 C2RY0J 50878551 Ki = 501.19 nM T77913 C1W6TV 50898777 Ki = 1258.93 nM T77913 CXMZ73 50898778 Ki > 10000 nM T77913 CX48AD 51002362 Ki = 586 nM T77913 C08FGN 51039225 Ki = 8.8 nM T77913 CS14BH 51039226 Ki = 4.9 nM T77913 CR70XF 51039227 Ki = 10.5 nM T77913 CE4KP1 51050257 Ki > 10000 nM T77913 CIJT81 51111982 Ki = 35 nM T77913 CF9V1U 52937018 Ki = 10 nM T77913 CS3BJ7 52937119 Ki = 6.31 nM T77913 C93QXP 52937222 Ki = 1 nM T77913 CPF7V0 52937223 Ki = 63.1 nM T77913 CYG24L 52937526 Ki = 0.1 nM T77913 CL8QZ3 52937527 Ki = 0.1585 nM T77913 CM36PE 52937629 Ki = 5.012 nM T77913 CRV61I 52937630 Ki = 0.3162 nM T77913 CEKB47 52937631 Ki = 0.1995 nM T77913 CZ0C5B 52937632 Ki = 398.11 nM T77913 CVX7U2 52937633 Ki = 630.96 nM T77913 C3ZX1Q 52937634 Ki > 1584.89 nM T77913 CY4N8T 52937728 Ki = 0.5012 nM T77913 C83WTP 52937729 Ki = 1.585 nM T77913 CQDS92 52937730 Ki = 1.995 nM T77913 CR0KW9 52937731 Ki = 0.7943 nM T77913 C2UV5S 52937732 Ki = 0.2512 nM T77913 C6XHP8 52937733 Ki = 1584.89 nM T77913 C3B5HN 52937734 Ki = 79.43 nM T77913 CK52QG 52937828 Ki = 31.62 nM T77913 CFV4D0 52937829 Ki = 1.585 nM T77913 C9MBQ2 52937830 Ki = 0.3162 nM T77913 C7OZN4 52944115 Ki = 3.981 nM T77913 CNQF49 52945978 Ki = 10 nM T77913 CRH43M 52946023 Ki = 64 nM T77913 CV2QJ5 52953079 IC50 = 530 nM T77913 CMJ62D 53245590 Ki = 1420 nM T77913 C7IMH5 53317594 Ki = 32 nM T77913 CT56HN 53317595 Ki = 249 nM T77913 CD0H8Z 53318872 Ki = 2.8 nM T77913 C90DGH 53318873 Ki = 162 nM T77913 C9MJ6C 53318874 Ki = 24.7 nM T77913 CWV40O 53320177 Ki = 7.2 nM T77913 CY5PO1 53320189 Ki = 4.3 nM T77913 C9JVY1 53321494 Ki = 24 nM T77913 CQ9PR5 53321511 Ki = 91 nM T77913 CW28NZ 53321512 Ki = 49 nM T77913 CSX14G 53321869 Ki > 10000 nM T77913 C9JUC1 53322838 Ki = 6.7 nM T77913 CEH78Z 53322839 Ki = 28 nM T77913 C78CYN 53322959 Ki = 13 nM T77913 C01OZU 53324167 Ki = 13.9 nM T77913 CR4W9L 53324553 Ki = 2376 nM T77913 C1WJH5 53325600 Ki = 48 nM T77913 CB37XF 53325861 Ki > 10000 nM T77913 CVNH56 53326712 Ki = 41 nM T77913 C4ZUJ9 53326724 Ki = 109 nM T77913 CU05TQ 53326725 Ki = 4605 nM T77913 C9Z3WY 53326726 Ki = 8.1 nM T77913 CE9NR7 53326727 Ki = 15.2 nM T77913 CLZ09P 53359025 Ki = 2372 nM T77913 CMOZ61 53475319 Ki = 110 nM T77913 CWH50X 53499206 Ki > 10000 nM T77913 C7HP2L 53524618 Ki > 10000 nM T77913 C9PQ6Y 53550713 Ki > 10000 nM T77913 C5Z1LN 54579956 IC50 = 610 nM T77913 C8BSR5 54579957 IC50 = 500 nM T77913 CSV05U 54580386 IC50 = 92 nM T77913 CJO04Z 54580942 IC50 = 120 nM T77913 CTN1V9 54580943 IC50 > 10000 nM T77913 C95ZWE 54581386 IC50 = 140 nM T77913 C7JB1W 54581387 IC50 = 135 nM T77913 C43JTB 54581997 IC50 = 390 nM T77913 CZ90MU 54581998 IC50 = 7160 nM T77913 CSW6I5 54581999 IC50 > 10000 nM T77913 CF2LE5 54582000 IC50 = 2790 nM T77913 C2QGE5 54582401 IC50 = 128 nM T77913 CPNO96 54582402 IC50 = 325 nM T77913 CWY0J9 54582938 IC50 = 4670 nM T77913 CGZ2A0 54582939 IC50 = 120 nM T77913 C63EMH 54582940 IC50 = 560 nM T77913 CA9UO3 54583384 IC50 = 128 nM T77913 CE2SJ4 54583938 IC50 = 320 nM T77913 CU97XI 54583939 IC50 = 7570 nM T77913 C8YV7J 54584335 IC50 = 540 nM T77913 C2TE0Z 54584885 IC50 > 10000 nM T77913 CM56LK 54585846 IC50 = 110 nM T77913 CNU5D7 54585847 IC50 = 220 nM T77913 C03QMG 54585848 IC50 = 1290 nM T77913 CTFW50 54586252 IC50 = 255 nM T77913 CP6B9G 54586253 IC50 = 150 nM T77913 C15SZR 54586254 IC50 = 54 nM T77913 C69IKU 54586255 IC50 = 75 nM T77913 CG37IB 54586256 IC50 = 63 nM T77913 C6SIO9 54586257 IC50 = 195 nM T77913 C39KWS 54586812 IC50 = 930 nM T77913 CY0G9U 54586813 IC50 = 650 nM T77913 C2WX4J 54587281 IC50 = 84 nM T77913 C5O6NT 54587282 IC50 = 153 nM T77913 CB72FX 54754351 Ki > 10000 nM T77913 CPS5V6 54764158 Ki > 10000 nM T77913 C2KG9D 56665110 Ki < 10000 nM T77913 CU0NE5 56672197 Ki < 10000 nM T77913 CP3L7E 56682094 Ki < 10000 nM T77913 CK9SG4 56781741 Ki = 2683 nM T77913 CY2S8M 56820088 Ki = 19 nM T77913 CY92VU 56835087 Ki > 10000 nM T77913 C0JMA7 56835088 Ki > 10000 nM T77913 C4E6HV 56835171 Ki = 10500 nM T77913 CJKO58 56852956 Ki = 724.44 nM T77913 CB0P9N 56944383 Ki = 69 nM T77913 C1TC7Q 56963799 Ki = 7055 nM T77913 C6H9UV 57345617 Ki = 1719 nM T77913 CZU6L2 57345618 Ki = 509 nM T77913 CK9G8H 57345619 Ki = 1247 nM T77913 C0P9VG 57390224 Ki = 776.25 nM T77913 CBD1F0 57390225 Ki = 457.09 nM T77913 CATM39 57390694 Ki = 665 nM T77913 C6S0IE 57390695 Ki = 129 nM T77913 C6SGK0 57391843 Ki = 16.6 nM T77913 CVO5M3 57393573 Ki = 4.9 nM T77913 CXV65K 57393730 Ki = 5.495 nM T77913 CADH19 57394285 Ki = 800.2 nM T77913 C01VOH 57395286 Ki = 5.7 nM T77913 CB09IO 57395287 Ki = 1 nM T77913 CI5M2U 57395620 Ki > 40000 nM T77913 CYC1Q5 57397055 Ki = 8.1 nM T77913 C25FTZ 57397056 Ki = 1.3 nM T77913 CE3U5Q 57397301 Ki = 100 nM T77913 C5D0RB 57398829 Ki = 6.3 nM T77913 CL4I6O 57398830 Ki = 1 nM T77913 C6N4KZ 57398985 Ki = 213.8 nM T77913 CJ41PW 57399432 Ki = 61 nM T77913 CR0BU6 57400501 Ki = 1 nM T77913 CE82XL 57400502 Ki = 1.9 nM T77913 CWZ50O 57400503 Ki = 1.3 nM T77913 C5MG6Q 57400504 Ki = 4 nM T77913 CJBU02 57400505 Ki = 1.4 nM T77913 C04XQW 57400700 Ki = 602.56 nM T77913 CZX05B 57401706 Ki = 212 nM T77913 C0MKN9 57402230 Ki = 92 nM T77913 C9D3ZE 57402314 Ki = 4.9 nM T77913 CXT2L1 57402315 Ki = 0.8 nM T77913 C4RN6L 57402471 Ki = 169.82 nM T77913 C6PH5T 57402472 Ki = 7.079 nM T77913 C0BWQ7 57402933 Ki = 2290.87 nM T77913 CX0B5M 57403525 Ki = 128.5 nM T77913 CWBG94 57403981 Ki = 187 nM T77913 C4RHF3 57404027 Ki > 10000 nM T77913 C49JDH 57404030 Ki = 1.2 nM T77913 C9SB1D 57404031 Ki = 24.6 nM T77913 CUOV05 57411066 Ki > 10000 nM T77913 CT89JH 57780007 Ki = 15.85 nM T77913 CT8RO7 57780008 Ki = 19.95 nM T77913 C5RIN4 57780016 Ki = 199.53 nM T77913 CE9WC0 57780017 Ki = 12.59 nM T77913 C1W4SB 57780018 Ki = 39.81 nM T77913 CT96WD 57780020 Ki = 12.59 nM T77913 C90EAP 59295914 Ki = 25.12 nM T77913 CFX9H8 59295925 Ki = 19.95 nM T77913 C5P6UI 59295926 Ki = 12.59 nM T77913 C18YQX 59295928 Ki = 63.1 nM T77913 C9NMZ2 59295931 Ki = 7.943 nM T77913 CV6PS4 59295935 Ki = 7.943 nM T77913 CA8T3Q 59295938 Ki = 10 nM T77913 C59QBR 59295939 Ki = 31.62 nM T77913 COG4S6 59295946 Ki = 50.12 nM T77913 CHP65R 59295958 Ki = 6.31 nM T77913 CRNJ03 59295960 Ki = 251.19 nM T77913 C3PCY5 59295968 Ki = 2.512 nM T77913 CYG56K 59295969 Ki = 5.012 nM T77913 C4PYU5 59295974 Ki = 50.12 nM T77913 CRZN12 59295978 Ki = 2.512 nM T77913 CR2T5D 59295982 Ki = 19.95 nM T77913 C4P3DW 59295984 Ki = 12.59 nM T77913 C17USX 59295994 Ki = 3.981 nM T77913 CJV58T 59296000 Ki = 19.95 nM T77913 C2K1TV 59296010 Ki = 6.31 nM T77913 C0KM5W 59296024 Ki = 63.1 nM T77913 CE73NG 59296033 Ki = 12.59 nM T77913 CT2P4Z 59296039 Ki = 63.1 nM T77913 C21AHO 59296041 Ki = 251.19 nM T77913 CXK7O5 59296048 Ki = 25.12 nM T77913 CF53RX 59296064 Ki = 19.95 nM T77913 CPE0B2 59296066 Ki = 10 nM T77913 C07OPL 59296073 Ki = 79.43 nM T77913 CFR8S7 59296077 Ki = 79.43 nM T77913 CMD56H 59296081 Ki = 2.512 nM T77913 C2HP9B 59296085 Ki = 100 nM T77913 CFCE90 59296090 Ki = 3.981 nM T77913 CGIL10 59296094 Ki = 125.89 nM T77913 C4H8KW 59296098 Ki = 501.19 nM T77913 CUC57E 59296099 Ki = 39.81 nM T77913 C1ZN0M 59296100 Ki = 25.12 nM T77913 CX6JS1 59296104 Ki = 3.981 nM T77913 CZW0V1 59296109 Ki = 199.53 nM T77913 C5TMB2 59296111 Ki = 15.85 nM T77913 CGF80H 59296114 Ki = 15.85 nM T77913 CQK9S3 59401826 Ki > 9300 nM T77913 C53BVH 59401876 Ki > 9300 nM T77913 CYKF93 59651916 Ki > 10000 nM T77913 CI5PM3 60165413 Ki = 52 nM T77913 C3K5JN 60165681 Ki = 46 nM T77913 CECR98 66615606 Ki = 501.19 nM T77913 CJ85YZ 66615617 Ki = 63.1 nM T77913 C9IQ1Y 66615619 Ki = 39.81 nM T77913 CFO03A 66615627 Ki = 31.62 nM T77913 CA59FS 66615678 Ki = 79.43 nM T77913 C9P6ZL 66615691 Ki = 199.53 nM T77913 C75RXH 66615702 Ki = 79.43 nM T77913 CL69HQ 66615705 Ki = 100 nM T77913 C7AZJ6 68168663 Ki = 1 nM T77913 CD3U6K 68731121 Ki > 10000 nM T77913 C6FZD0 68846936 Ki = 63.1 nM T77913 CZPM30 68849581 Ki = 100 nM T77913 C5PY2V 68938028 Ki = 31.62 nM T77913 C6IP8Q 69082816 Ki = 7010 nM T77913 C07YOG 69260079 Ki = 10 nM T77913 CV7P3D 69260851 Ki = 63.1 nM T77913 C4QO7E 69260946 Ki = 5.012 nM T77913 CO9U3M 69262172 Ki = 6.31 nM T77913 C7HN5L 69272932 Ki = 15.85 nM T77913 CJ2D3I 69274365 Ki = 5.012 nM T77913 C5FAB3 69314950 Ki = 3.5 nM T77913 COD5Y1 69347575 Ki = 100 nM T77913 C51DQR 69347707 Ki = 125.89 nM T77913 C8F1CY 69347719 Ki = 63.1 nM T77913 C93COF 69347980 Ki = 50.12 nM T77913 CPW42A 69348078 Ki = 25.12 nM T77913 CH3SB0 69355600 Ki = 3890.45 nM T77913 CZO27L 69826668 Ki = 25.12 nM T77913 C18RLK 71072034 Ki = 100 nM T77913 C4C0SP 71072040 Ki = 50.12 nM T77913 C1YNH6 71072044 Ki = 50.12 nM T77913 CVU3G7 71072050 Ki = 50.12 nM T77913 C2M1JY 71072052 Ki = 15.85 nM T77913 CE6Y8Z 71072057 Ki = 125.89 nM T77913 C0Z3KN 71072081 Ki = 15.85 nM T77913 C3FR6X 71072104 Ki = 63.1 nM T77913 C1BEC9 71072113 Ki = 79.43 nM T77913 CNY09L 71072115 Ki = 25.12 nM T77913 CFNZ23 71072118 Ki = 50.12 nM T77913 CC43QK 71151588 Ki = 160 nM T77913 C6QYO1 71449142 Ki = 446.68 nM T77913 CBQ8P4 71449250 Ki = 0.6918 nM T77913 CH5X6M 71449584 Ki = 15.85 nM T77913 CH5PX8 71449585 Ki = 5.012 nM T77913 CUKW48 71449857 Ki = 25.12 nM T77913 COVR94 71449858 Ki = 79.43 nM T77913 C5M7WE 71449859 Ki = 39.81 nM T77913 CV28YI 71450058 Ki = 20 nM T77913 C9VZ8J 71450550 Ki = 3727 nM T77913 CE6YD5 71450707 Ki > 10000 nM T77913 CSYN25 71450777 Ki = 12.59 nM T77913 CDI84E 71450922 IC50 > 10000 nM T77913 CB83YL 71451044 Ki = 0.631 nM T77913 C3FC1H 71451390 Ki = 398.11 nM T77913 C4W6YG 71451391 Ki = 158.49 nM T77913 CI65MW 71451392 Ki = 100 nM T77913 C9OG2Q 71451671 Ki = 15.85 nM T77913 C4TWS5 71452172 Ki > 10000 nM T77913 C4NDR3 71452382 Ki = 3839 nM T77913 CE1Z0V 71452601 Ki = 0.3162 nM T77913 C59WFT 71452602 Ki = 501.19 nM T77913 CP45AB 71452695 Ki = 20000 nM T77913 C0YXD3 71452871 Ki = 0.2512 nM T77913 CY7NM9 71452872 Ki = 0.3548 nM T77913 C8C9JT 71453204 Ki = 100 nM T77913 CB86VX 71453505 Ki = 25.12 nM T77913 C4X9KY 71454294 Ki = 6500 nM T77913 CA65OQ 71454295 Ki = 1000 nM T77913 C02FKR 71454296 Ki = 5.012 nM T77913 CZ8W9G 71454365 Ki = 316.23 nM T77913 C4JN5I 71454639 Ki = 0.631 nM T77913 CB6PF0 71455217 Ki = 31.62 nM T77913 CD4HQ6 71456045 Ki = 1400 nM T77913 CD78KL 71456046 Ki = 2600 nM T77913 CMBU21 71456359 Ki = 0.5129 nM T77913 CVT39B 71456360 Ki = 1 nM T77913 CK87DI 71456361 Ki = 1.288 nM T77913 CL9BS3 71456722 Ki = 79.43 nM T77913 CT0OQ6 71456725 Ki = 19.95 nM T77913 CIXY68 71457009 Ki > 6309.57 nM T77913 CGP6K8 71457010 Ki = 50.12 nM T77913 C7MNB5 71457264 Ki = 681.8 nM T77913 CSX5J0 71457844 Ki = 5500 nM T77913 C3VMS0 71458203 Ki = 0.3467 nM T77913 C8T5EJ 71458204 Ki = 0.3162 nM T77913 CZ6BX7 71458205 Ki = 0.537 nM T77913 CZW7X0 71458868 Ki = 19.95 nM T77913 CHC0Z2 71458869 Ki = 100 nM T77913 CF1PV0 71458870 Ki > 5011.87 nM T77913 CK5T4P 71459604 Ki = 8858 nM T77913 CD10CQ 71459761 Ki = 490 nM T77913 CJ1M6I 71459762 Ki = 12.59 nM T77913 CMI1A6 71459825 Ki = 501.19 nM T77913 CP26GF 71460416 Ki = 63.1 nM T77913 CH51UB 71460419 Ki = 31.62 nM T77913 C1GV6P 71461541 Ki = 1258.93 nM T77913 CEBC62 71461781 Ki = 0.912 nM T77913 C9DJ1V 71461782 Ki = 0.3981 nM T77913 C9UG2X 71462100 Ki = 50.12 nM T77913 CYM4X2 71462102 Ki = 19.95 nM T77913 CL4MZ5 71462103 Ki = 39.81 nM T77913 CX97KJ 71462389 Ki = 125.89 nM T77913 C6UBQ4 71462390 Ki = 31.62 nM T77913 CQ36LR 71462391 Ki = 199.53 nM T77913 C5CS7I 71463287 Ki = 3.162 nM T77913 C05HIC 71463288 Ki = 19.95 nM T77913 CLQ31I 71519674 Ki = 20892.96 nM T77913 CRM9Q1 71525678 Ki = 33884.42 nM T77913 C2GK7O 71525679 Ki = 11220.18 nM T77913 C8A0NC 71525681 Ki = 16595.87 nM T77913 CE92DF 71528209 Ki = 1662 nM T77913 CI0GU8 71660496 IC50 > 48500 nM T77913 C93WIJ 71712245 Ki = 10471.29 nM T77913 C90EXP 71723301 Ki = 19.95 nM T77913 CF01OQ 71937057 Ki = 44 nM T77913 C0PSF9 72138721 Ki = 134 nM T77913 CR3Z1P 72152555 Ki = 32 nM T77913 C24ZSV 72152556 Ki = 302 nM T77913 CWT8O4 72152557 Ki = 40 nM T77913 CZ49CG 72152558 Ki = 2455 nM T77913 CWH6T3 72548703 IC50 = 1.7 nM T77913 CC6Q5R 72771081 Ki < 100 nM T77913 CC65OA 73213195 Ki = 47.86 nM T77913 CW83DK 73213196 Ki > 10000 nM T77913 CCV91B 73346042 Ki = 512 nM T77913 CR97NO 73347825 Ki = 1359 nM T77913 CC35AI 73347827 Ki > 10000 nM T77913 CW8A0Y 73349359 Ki = 5569 nM T77913 C1NJ0R 73353884 Ki = 4178 nM T77913 C4F7VK 73355415 Ki = 4736 nM T77913 CAI63V 73355417 Ki > 10000 nM T77913 C2E7QW 75201901 IC50 = 4600 nM T77913 C8IDL3 75306277 Ki = 3.162 nM T77913 CT64PM 76317221 Ki > 2511.89 nM T77913 C28RIZ 76518514 Ki = 1719 nM T77913 CQ7W3I 89474811 Ki = 3.162 nM T77913 CF05GE 90654501 Ki = 29512.09 nM T77913 C1BJC6 90654502 Ki = 31622.78 nM T77913 CPY4X2 90654503 Ki = 2238.72 nM T77913 C0J5YH 91864602 Ki = 597 nM T77913 CRX16J 91884611 IC50 = 177 nM T77913 CLR87F 94496003 Ki = 1144 nM T77913 CNUM64 95104704 Ki = 718 nM T77913 CK83CL 95198280 Ki = 1866 nM T77913 CMG1N3 95214051 Ki = 2562 nM T77913 C5GJA7 95232163 Ki = 4241 nM T77913 C8QJW7 95338888 Ki = 310 nM T77913 C0BAG2 95339350 Ki = 1110 nM T77913 C4BRK3 95339542 Ki = 322 nM T77913 CFA3D4 112936251 Ki = 1122.02 nM T77913 C85IFK 112936262 Ki = 5248.07 nM T77913 CLQ10U 112936267 Ki = 3311.31 nM T77913 C5DU3L 112936341 Ki = 2511.89 nM T77913 C1LO3K 112936352 Ki = 4168.69 nM T77913 CI0DB6 112936357 Ki = 1949.84 nM T77913 CSB25E 118709750 Ki = 1207 nM T77913 CD4S9R 118709751 Ki = 1009 nM T77913 C2K6ML 118721928 Ki = 153 nM T77913 C6YF0A 118721929 Ki = 289 nM T77913 CK03VE 118721930 Ki = 147 nM T77913 CBM7V0 118721934 Ki = 4647 nM T77913 C4G3YC 118734875 Ki > 10000 nM T77913 C9AIE1 118734876 Ki > 10000 nM T77913 CK61AT 127026016 Ki = 1905.46 nM T77913 C9LJH1 127026017 Ki = 1071.52 nM T77913 C3QBS9 127026018 Ki = 1862.09 nM T77913 CDF56P 127026019 Ki = 1174.9 nM T77913 CTBN56 127026052 Ki = 79.43 nM T77913 CQ0ZT9 127035062 Ki = 1297 nM T77913 C0Z9RT 127035835 Ki = 2089.3 nM T77913 C20IYZ 127035836 Ki = 3388.44 nM T77913 CL9PN3 127035837 Ki = 1949.84 nM T77913 CU49VE 127036186 Ki = 676.08 nM T77913 CG06BD 127036932 Ki = 100 nM T77913 CVW71O 127036953 Ki = 100 nM T77913 CST95G 127036978 Ki = 5754.4 nM T77913 CIK1S7 127036979 Ki = 9332.54 nM T77913 C1ICF6 127036980 Ki = 891.25 nM T77913 CP6IZ7 127036981 Ki = 8128.31 nM T77913 CY6T9R 127036982 Ki = 6309.57 nM T77913 C4KO0Z 127048828 Ki = 8750 nM T77913 C2XT3K 127048890 Ki > 10000 nM T77913 CC7BU0 127049059 Ki = 535 nM T77913 C42FHY 127049060 Ki = 273 nM T77913 CY38PR 127049156 Ki > 10000 nM T77913 CG35RK 127049855 Ki = 7910 nM T77913 C5BZ6T 127049856 Ki = 6780 nM T77913 CZS1L6 127049862 IC50 = 2560 nM T77913 CZD91J 127049863 IC50 = 972 nM T77913 CF0Y6S 127050431 Ki > 10000 nM T77913 CX53AC 127050632 Ki = 263 nM T77913 CF3BH2 127050775 Ki > 10000 nM T77913 C5P1EB 127050776 Ki > 10000 nM T77913 CH8G4Z 127051047 Ki > 10000 nM T77913 CH8Y7R 127051301 Ki > 10000 nM T77913 CTL0S1 127051516 Ki = 1.175 nM T77913 CTL8J1 127051843 Ki = 158.49 nM T77913 CF6V9Q 127051844 Ki = 1427 nM T77913 C8TNB1 127051845 Ki = 199.53 nM T77913 C5ONG1 127051864 Ki = 186.21 nM T77913 CVQW26 127051865 Ki = 1023.29 nM T77913 CB25IM 127051958 Ki > 10000 nM T77913 CNR4Q9 127051986 Ki > 10000 nM T77913 C3YSF2 127052292 Ki = 9350 nM T77913 C9OSN3 127052293 Ki = 6080 nM T77913 C3WA2L 127052294 Ki = 3050 nM T77913 CYWZ45 127052295 Ki > 10000 nM T77913 CK1IF9 127052296 Ki > 10000 nM T77913 CHJE58 127052297 Ki > 10000 nM T77913 CCY71I 127052465 Ki = 3630.78 nM T77913 C2E9VX 127052467 Ki = 831.76 nM T77913 CSQ2N8 127052486 Ki = 501.19 nM T77913 C4YJ8H 127052487 Ki = 245.47 nM T77913 C98YAI 127052634 Ki > 10000 nM T77913 C7T4VH 127052635 Ki = 8350 nM T77913 CLU7C1 127052757 Ki = 738 nM T77913 C95KYT 127052758 Ki = 380.19 nM T77913 C6GC0F 129186534 IC50 = 123 nM T77913 C8KM6N 129186554 IC50 = 127 nM T77913 CEZT92 129186564 IC50 = 162 nM T77913 C50GOC 130442480 Ki > 10000 nM T77913 CM04RF 130442572 Ki = 9800 nM T77913 CS58HX 132060734 Ki = 298 nM T77913 CY8B9L 132060743 Ki = 483 nM T77913 C4VNA6 132060746 Ki = 594 nM T77913 C4OC0I 132060752 Ki = 1061 nM T77913 C7FM0U 132060763 Ki = 869 nM T77913 CGHO19 132060770 Ki = 62 nM T77913 CT81OY 132060776 Ki = 336 nM T77913 C7CSU4 132075278 Ki = 1739 nM T77913 CAVB41 132584404 Ki > 10000 nM T77913 C8O2EP 134130246 Ki = 812.83 nM T77913 C8X4FV 134132468 Ki = 6.31 nM T77913 CQX4U3 134133064 Ki = 3867 nM T77913 CQ95LB 134133571 Ki > 2511.89 nM T77913 C0J2ML 134133604 Ki = 549.54 nM T77913 CP0E5M 134133632 Ki = 998 nM T77913 CM0TS6 134133967 Ki = 293 nM T77913 CR0JY2 134134674 Ki = 2.512 nM T77913 CYLO91 134135965 Ki = 1.995 nM T77913 CG9J7V 134136763 Ki = 15.85 nM T77913 C3W5SM 134139893 Ki = 79.43 nM T77913 CHG9Z5 134140686 Ki > 2511.89 nM T77913 C5HSW6 134141284 Ki = 12.59 nM T77913 CLW86T 134141354 Ki = 3162.28 nM T77913 CFW7E3 134141385 Ki > 2511.89 nM T77913 CU5JS4 134142911 Ki = 1584.89 nM T77913 C24FED 134142976 Ki = 1584.89 nM T77913 C3NT1H 134143679 Ki = 251.19 nM T77913 C2IM4X 134143913 Ki = 1000 nM T77913 CR5L4K 134144303 Ki = 1000 nM T77913 CF23UV 134144915 Ki = 100 nM T77913 CW7OG9 134145047 Ki = 3.162 nM T77913 C73XEV 134145497 Ki = 63.1 nM T77913 CFTA36 134145956 Ki = 25.12 nM T77913 CC9P2T 134146194 Ki = 268 nM T77913 CBU81N 134149168 Ki > 10000 nM T77913 C4UG2X 134150352 Ki = 31.62 nM T77913 C1PQ5T 134150412 Ki = 398.11 nM T77913 CLU34D 134151427 Ki = 24 nM T77913 CV3AK8 134151839 Ki = 19.95 nM T77913 CK2UY5 134152174 Ki = 15.85 nM T77913 CB6M5Y 134153538 Ki = 560 nM T77913 C79TEI 134154068 Ki = 245.47 nM T77913 CMJ1U3 134154387 Ki = 1437 nM T77913 C4VGJ5 134154679 Ki = 323.59 nM T77913 C79QLN 134155460 Ki = 290 nM T77913 CY5S3R 134155594 Ki = 6.31 nM T77913 CLC9U1 134156932 Ki = 316.23 nM T77913 C08AQK 134156987 Ki = 7.943 nM T77913 CF32WY 134157080 Ki = 251.19 nM T77913 C1GY2T 135156251 EC50 > 10000 nM T77913 C2PT4I 135356876 Ki = 170 nM T77913 C5OU1T 135409492 Ki = 87 nM T77913 C9B7XA 135458410 Ki = 18.3 nM T77913 C4PM9W 135515431 Ki = 6 nM T77913 CE40DG 135882460 Ki > 10000 nM T77913 C5KE3N 135986088 Ki = 190 nM T77913 CBS93O 136030655 Ki > 10000 nM T77913 C8I7CO 136141537 Ki > 10000 nM T77913 C37YXA 136152971 Ki = 2.6 nM T77913 CRH19Y 136192874 Ki > 1000 nM T77913 C56FVS 136192886 Ki > 10000 nM T77913 C78RFZ 136229178 Ki = 15.85 nM T77913 C63FEC 137125241 IC50 > 30000 nM T77913 CIHJ46 137125256 IC50 = 1 nM T77913 CPCY48 137645406 Ki = 8 nM T77913 CPI68E 137646281 Ki = 40 nM T77913 C04XYN 137653567 IC50 = 132 nM T77913 C85BSY 145963127 Ki > 10000 nM T77913 CEN94V 145963961 IC50 = 923 nM T77913 C1B8QW 145964299 IC50 = 4420 nM T77913 CLM10C 145966333 IC50 = 418 nM T77913 C8I7QL 145980875 Ki = 718 nM T77913 C1DW4U 145983928 IC50 = 195 nM T77913 CNJH37 145986752 Ki = 7031 nM T77913 CUGO10 145988693 Ki = 814 nM T77913 CMJ46R 145990794 IC50 = 174 nM T77913 CCP2U1 145992489 Ki = 718 nM T77913 C9PS8N 145993117 IC50 = 253 nM T77913 C0Z6YX 145993493 IC50 = 305 nM T77913 CC2G1V 146025727 Ki = 2600 nM T77913 CI50EP 147863431 IC50 = 6.23 nM T77913 CMQ7G1 148123909 IC50 = 52.85 nM T77913 C1PJL8 149227688 IC50 = 36.71 nM T77913 C2HU8I 150575506 IC50 = 9.28 nM T77913 C6P3SR 153287553 Ki > 10000 nM T77913 CV9G7Z 153287572 Ki > 10000 nM T77913 CO85KL 153287574 Ki > 10000 nM T77913 C4BQ2D 155515934 Ki = 3.162 nM T77913 C5LNQ4 155518920 IC50 = 2.95 nM T77913 CIQ68C 155519275 Ki = 0.631 nM T77913 CUSA24 155519891 Ki > 10000 nM T77913 CV0H6F 155521446 Ki = 5.012 nM T77913 C85VUB 155522480 IC50 = 8.14 nM T77913 C62VSP 155523802 Ki = 3.981 nM T77913 CPB1Q0 155526952 IC50 = 40.22 nM T77913 CIW73O 155527187 Ki = 7.943 nM T77913 CIDA50 155532375 IC50 = 4.56 nM T77913 CB79ZW 155536080 Ki = 3162.28 nM T77913 CTK09Y 155536195 IC50 = 17.65 nM T77913 C20KGT 155536963 Ki = 1.259 nM T77913 CYV64X 155537274 Ki = 3.981 nM T77913 C7V4EF 155539495 Ki = 1.778 nM T77913 C5H1UA 155541322 IC50 = 20.98 nM T77913 CGP4Z6 155544367 IC50 = 4160 nM T77913 CF92LJ 155545274 IC50 = 81.78 nM T77913 C6H0AR 155545724 IC50 = 27.88 nM T77913 CBV8E3 155549599 IC50 = 8.9 nM T77913 CIJ06P 155549722 IC50 = 28.41 nM T77913 C1RLI0 155553370 Ki > 10000 nM T77913 C70AUP 155554175 IC50 = 11.97 nM T77913 CXEQ70 155555597 Ki = 0.3981 nM T77913 CFBK91 155556183 Ki = 2.512 nM T77913 CS86UH 155557098 IC50 = 4.74 nM T77913 CFKB62 155561547 Ki = 2.138 nM T77913 C8HR4Q 155567029 Ki = 1270 nM T77913 C2EI0V 155567448 Ki = 3.162 nM T77913 C2YO5R 155567541 Ki = 0.7943 nM T77913 C8AM0E 155568607 IC50 = 3.67 nM T77913 C3N9VU 10251906 Ki = 189 nM T77913 CP9TR0 10324985 Ki = 150 nM T77913 CB2VD8 44241743 Ki > 1000 nM T77913 D01CXD 10398175 Ki = 197 nM T77913 D01HJZ 83632 Ki = 5172 nM T77913 D01JXM 46222048 Ki > 1000 nM T77913 D02GNN 119812 Ki = 64 nM T77913 D02HNQ 46182736 IC50 > 10000 nM T77913 D02SDX 151221 Ki = 75 nM T77913 D02SQF 37463 EC50 = 15848.93 nM T77913 D02YSX 197033 IC50 = 160 nM T77913 D03SNI 24759623 Ki = 741.31 nM T77913 D03VUU 44521012 Ki = 48 nM T77913 D04SCQ 3015863 Ki = 1670 nM T77913 D04TPO 16006492 Ki = 1100 nM T77913 D04TWX 9794475 Ki > 2000 nM T77913 D05BYD 9906860 Ki = 69183.1 nM T77913 D05KUM 135446209 Ki = 22 nM T77913 D05RGW 11313837 Ki < 10000 nM T77913 D05RKS 20293994 Ki = 386 nM T77913 D05YFZ 44373221 Ki = 137 nM T77913 D05ZUX 44207909 Ki = 780 nM T77913 D07RYR 44396235 Ki = 15.85 nM T77913 D08RCH 44566054 IC50 = 3600 nM T77913 D08TBU 15723 Ki = 659 nM T77913 D09RPR 16737207 Ki > 10000 nM T77913 D0A1DE 10917690 IC50 = 59 nM T77913 D0B0PP 79698 Ki = 2758 nM T77913 D0BT1A 75919 IC50 = 1258.93 nM T77913 D0C7FL 77575 Ki > 10000 nM T77913 D0D3YN 1238 Ki = 0.19 nM T77913 D0D8GV 9830741 Ki = 54 nM T77913 D0E1RX 11335419 Ki = 10 nM T77913 D0E9SR 4908365 Ki = 977.24 nM T77913 D0F0IA 11301655 Ki > 2000 nM T77913 D0FF6S 16038374 IC50 > 10000 nM T77913 D0FU5E 10220053 Ki > 1000 nM T77913 D0G6AQ 23786499 EC50 = 199.53 nM T77913 D0H3DY 10374457 EC50 = 864 nM T77913 D0H4TP 9798547 Ki > 2511.89 nM T77913 D0H8XV 12963076 Ki = 0.4 nM T77913 D0I0UW 45485498 Ki = 3200 nM T77913 D0I3XA 6422124 Ki > 2511.89 nM T77913 D0I5CT 126688 EC50 = 15848.93 nM T77913 D0J6XO 9884746 Ki = 1905.46 nM T77913 D0KK4C 10154137 EC50 > 0.0001 nM T77913 D0L5MW 181743 Ki > 10000 nM T77913 D0M9IC 441082 Ki > 10000 nM T77913 D0PN9R 16655023 Ki = 74 nM T77913 D0R8UU 44396220 Ki = 25.12 nM T77913 D0RG8O 10447834 IC50 = 794.33 nM T77913 D0S0WX 10354158 Ki = 175 nM T77913 D0S3WR 120445 Ki = 70 nM T77913 D0SQ0T 10942498 EC50 > 0.0001 nM T77913 D0T2RY 9948320 Ki = 610 nM T77913 D0T7AR 14827778 IC50 = 1995.26 nM T77913 D0TC5E 91613 EC50 = 794.33 nM T68834 D0G2MW 446284 IC50 = 2000 nM T68834 D0O1TC 5280581 IC50 = 2000 nM T68834 D0Q5XX 445580 IC50 = 2000 nM T68834 C3PAY7 5312529 IC50 = 2000 nM T68834 CE4UQ7 10544716 IC50 = 2500 nM T68834 C2GHN3 11279751 EC50 > 100000 nM T68834 CB0QA4 14164519 IC50 > 30000 nM T68834 C3M1DV 24822699 EC50 > 100000 nM T68834 CYIV49 44378315 EC50 = 1540 nM T68834 CUJ54O 49778909 IC50 = 6 nM T68834 CGR05H 49800284 IC50 = 2150 nM T68834 C2AN3Y 49800286 IC50 = 11000 nM T68834 C5T9BE 49800558 IC50 = 700 nM T68834 CCF5O6 49800560 IC50 = 570 nM T68834 CY8PX3 49800561 IC50 = 13700 nM T68834 CT0H3S 49800562 IC50 = 11770 nM T68834 C6IE2K 49800564 IC50 = 17670 nM T68834 C57ZQX 49800839 IC50 = 18000 nM T68834 CKE4A1 49800841 IC50 = 750 nM T68834 CNES29 49800843 IC50 = 1630 nM T68834 C8RP2B 49801419 IC50 = 566 nM T68834 C7TMZ9 49802026 IC50 = 2.7 nM T68834 CZ61BN 49802029 IC50 = 2175 nM T68834 CU01JQ 49802030 IC50 > 30000 nM T68834 C6YKX3 49802316 IC50 = 2.2 nM T68834 C58WZX 49802318 IC50 = 1120 nM T68834 C32RUD 49802589 IC50 = 81 nM T68834 C9KH6D 49804576 IC50 = 1130 nM T68834 CF24AR 49804577 IC50 = 90 nM T68834 CA7DO3 49804580 IC50 = 6060 nM T68834 CD2L9F 49804581 IC50 = 314 nM T68834 C6Y7NZ 49804582 IC50 = 20680 nM T68834 CB6XR5 53248990 IC50 = 7.5 nM T68834 CZ4J2U 66644000 IC50 = 9750 nM T68834 CY68KJ 66644017 IC50 = 141 nM T68834 CP9H7E 66644128 IC50 = 16 nM T68834 CS02HE 66644266 IC50 = 4030 nM T68834 CC89EN 68036050 IC50 = 550 nM T68834 C3X2MH 68751567 IC50 > 30000 nM T68834 CSPL78 71717596 IC50 = 1170 nM T68834 CA21HM 71720638 IC50 = 400 nM T68834 CB59JD 76317856 IC50 = 26 nM T68834 CYJW96 76328737 IC50 = 30 nM T68834 CY0QC5 76332419 IC50 = 323 nM T68834 CW9IR7 76336045 IC50 = 136 nM T68834 C4A9FP 76336046 IC50 = 638 nM T68834 C1E4DL 102164179 EC50 = 380 nM T68834 C2H7VC 118707104 IC50 = 18500 nM T68834 CTBQ09 118707105 IC50 = 460 nM T68834 CTLJ19 122588209 IC50 = 11 nM T68834 C5PUS9 122588230 IC50 = 0.28 nM T68834 CI07RE 122588268 IC50 = 223 nM T68834 CA5M1T 122588275 IC50 = 0.12 nM T68834 C8DOL3 122600340 IC50 = 38 nM T68834 CP6WV5 122600362 IC50 = 23 nM T68834 CCK82Q 137638047 IC50 = 1330 nM T68834 CD65JH 137638887 IC50 = 8150 nM T68834 CIL21A 137644937 IC50 = 1360 nM T68834 CR7W9B 137645745 IC50 = 580 nM T68834 CMWV08 137647550 IC50 = 23 nM T68834 C7LJ3D 137655326 IC50 = 720 nM T68834 C18GSA 137655720 IC50 = 5500 nM T68834 C5QIL7 137660364 IC50 = 4060 nM T68834 CU20KQ 145962053 EC50 = 2080 nM T68834 CGR1O4 145979016 IC50 = 210 nM T68834 CN63FR 145979967 IC50 = 2.1 nM T68834 CG3YT6 145980814 IC50 = 0.38 nM T68834 CU8B6E 145982307 IC50 = 38 nM T68834 CSMQ31 145984923 IC50 = 120 nM T68834 C8D5TM 145984927 IC50 = 12 nM T68834 CSZ8J9 145986668 IC50 = 18 nM T68834 CM4V3S 145989845 IC50 = 750 nM T68834 C86GOS 145993055 IC50 = 260 nM T68834 D0D2MN 10568747 IC50 = 500 nM T68834 D0JH4U 6438757 EC50 = 56 nM T68834 D0US4S 5283159 EC50 = 7 nM T68834 D0Z5QA 5283155 IC50 = 500 nM T94627 D06IAR 60961 Ki = 5300 nM T94627 D0TS1Z 5790 IC50 > 1000000 nM T94627 D0Y7DP 6029 Ki = 31000 nM T94627 D00YSJ 158795 Ki = 231000 nM T94627 CM2NR3 676310 IC50 > 1000000 nM T94627 CQUE70 11168331 IC50 = 62 nM T94627 C80VJG 11544329 IC50 > 100000 nM T94627 CU5K3A 11604803 IC50 = 1500 nM T94627 C5DVI4 11613505 IC50 = 940 nM T94627 C43FDR 11953391 IC50 > 100000 nM T94627 CO2UW0 13965968 IC50 = 52000 nM T94627 CP53KE 22803321 IC50 > 100000 nM T94627 CQDS54 46887269 IC50 > 100000 nM T94627 CTQW91 54553601 IC50 = 289000 nM T94627 C7MR1H 56975630 IC50 > 100000 nM T94627 C6ACJ2 59034940 IC50 = 233000 nM T94627 CD9PV3 59035027 IC50 = 536000 nM T94627 CK98IV 59035037 IC50 = 5700 nM T94627 CX9P4M 59460356 IC50 = 10400 nM T94627 C30KQD 59460362 IC50 = 1000 nM T94627 CR5JW7 59460372 IC50 = 1600 nM T94627 C4AF5O 59460394 IC50 = 1200 nM T94627 CFN93G 59460406 IC50 = 1300 nM T94627 CFQJ18 59460412 IC50 = 2300 nM T94627 C3Q5DG 59460418 IC50 = 5400 nM T94627 CSL7X3 59460423 IC50 = 5300 nM T94627 C69MXA 59460440 IC50 = 2700 nM T94627 C0K4UL 59460453 IC50 = 5500 nM T94627 C1QK9F 59460466 IC50 = 1100 nM T94627 C9GVC8 59460469 IC50 = 3100 nM T94627 C0F4PD 59460471 IC50 = 1300 nM T94627 CL0VD3 59460477 IC50 = 3300 nM T94627 CYM17L 59460487 IC50 = 1100 nM T94627 C9GNY1 59460512 IC50 = 5200 nM T94627 CU0CL5 118737953 IC50 = 65000 nM T94627 C3JBR0 118737954 IC50 = 19000 nM T94627 C4NQC9 118737955 IC50 = 11000 nM T94627 C96MYH 118737956 IC50 = 5700 nM T94627 CVHB32 118737957 IC50 = 5400 nM T94627 C79VFI 118737958 IC50 = 11000 nM T94627 C9QT6N 118737959 IC50 > 100000 nM T94627 C7IHE6 118737960 IC50 = 13000 nM T94627 C0B9IG 118737961 IC50 = 36000 nM T94627 C3EU0H 118737962 IC50 > 100000 nM T94627 CT5Z6D 118737963 IC50 = 21000 nM T94627 CZ5OF6 118737964 IC50 > 100000 nM T94627 C7PD5K 118737965 IC50 > 100000 nM T94627 CJH19M 118737966 IC50 > 100000 nM T94627 C5Z8OQ 118737967 IC50 > 100000 nM T94627 CN0OH9 118737968 IC50 > 100000 nM T94627 CAU2B9 118737969 IC50 > 100000 nM T94627 CTH0G3 118737970 IC50 > 100000 nM T94627 CT49BF 127045051 IC50 = 9300 nM T94627 C9KP4Z 135966733 IC50 = 20100 nM T94627 D05TGQ 59460354 IC50 = 640 nM T94627 D06WAL 6072 IC50 = 100000 nM T14380 D0U5GB 92727 IC50 > 20000 nM T14380 D0ZU9R 392622 IC50 > 20000 nM T14380 CI81AL 44530662 IC50 = 977 nM T14380 C97WEM 75593288 IC50 = 19 nM T14380 C6PYO2 85470898 IC50 = 0.2 nM T14380 CY9G8O 118716198 IC50 = 774 nM T14380 CL6TE3 118716321 IC50 = 378 nM T14380 C4IZ7G 118716325 IC50 = 625 nM T14380 CQB1N2 118716328 IC50 = 550 nM T14380 CEU78H 118717559 IC50 = 556 nM T14380 CCT87K 118717561 IC50 = 613 nM T14380 CYR34C 118717562 IC50 = 865 nM T14380 C3U5OB 118717564 IC50 = 967 nM T14380 CSWB75 118717566 IC50 > 20000 nM T14380 C4FWD7 118717568 IC50 > 20000 nM T14380 CH87TO 118717570 IC50 = 614 nM T14380 CVU1N5 118717571 IC50 > 20000 nM T14380 CXAF54 118717573 IC50 > 20000 nM T14380 CBO59G 118717574 IC50 > 20000 nM T14380 CH2WP5 118717577 IC50 > 20000 nM T14380 CWL05M 118717579 IC50 > 20000 nM T14380 C6VM8P 118717581 IC50 > 20000 nM T14380 CVKR02 118717582 IC50 = 29 nM T14380 C5SZC4 118717584 IC50 = 26 nM T14380 C50AUM 118717586 IC50 = 77 nM T14380 CHNF21 118717648 IC50 = 230 nM T14380 C98MHD 118717651 IC50 = 530 nM T14380 C1UGM6 118717653 IC50 = 622 nM T14380 CMV83O 118717655 IC50 = 772 nM T14380 CS0T9I 118717657 IC50 = 569 nM T14380 C1BX8S 118717659 IC50 = 300 nM T14380 C64WVI 118717661 IC50 = 2010 nM T14380 CE10FR 122206045 IC50 = 26 nM T14380 CFX1M8 127032622 IC50 = 0.8 nM T14380 C5L8DM 127034977 IC50 = 48000 nM T14380 CIOM15 127034978 IC50 = 890 nM T14380 CU47OV 127035290 IC50 > 50000 nM T14380 CBJ90V 127036340 IC50 = 15600 nM T25637 D0X5SD 3117 IC50 = 150 nM T25637 C49BCY 1570 IC50 = 18000 nM T25637 CZ7IA3 1647 IC50 = 73 nM T25637 C72PUR 7504 IC50 = 64700 nM T25637 C5FC8N 29147 IC50 = 719 nM T25637 CRWQ75 67326 IC50 = 26000 nM T25637 C83DJV 77317 IC50 = 1220 nM T25637 C04SFY 82608 IC50 = 670 nM T25637 C64RIA 83275 IC50 = 8210 nM T25637 CKC31Q 86633 IC50 = 2100 nM T25637 C4ZB8R 245718 IC50 > 100000 nM T25637 C8WZ4I 427814 IC50 = 47000 nM T25637 CU3F0X 571728 IC50 = 3620 nM T25637 C39MKT 712750 IC50 = 25000 nM T25637 COB3T1 2132963 IC50 > 100000 nM T25637 C0N9OQ 2756472 IC50 = 4970 nM T25637 C1CNZ9 2756474 IC50 = 1110 nM T25637 CF2N8O 2794167 IC50 = 126 nM T25637 C41QRG 2794826 IC50 = 3540 nM T25637 C94LDM 6459851 IC50 = 45000 nM T25637 CKEY45 10606883 IC50 = 35000 nM T25637 C3J2IR 12017326 IC50 = 6040 nM T25637 CPIV30 13194096 IC50 = 75000 nM T25637 CW1FA3 16227983 IC50 = 1200 nM T25637 CBZP95 16780874 IC50 = 1800 nM T25637 C8E2GN 16782615 IC50 = 203 nM T25637 CAQP19 16785630 IC50 = 309 nM T25637 CXV21M 21066395 IC50 = 902 nM T25637 C09ALD 22958840 IC50 > 100000 nM T25637 CKP0U7 23160415 IC50 = 385 nM T25637 CMO3B7 29130197 IC50 = 7800 nM T25637 CC9VJ0 39047495 IC50 = 3800 nM T25637 C10ECH 45480462 IC50 = 431 nM T25637 COVQ63 55265285 IC50 = 999 nM T25637 C3PTZ7 70700688 IC50 = 1000 nM T25637 CPG73S 73417116 IC50 > 100000 nM T25637 CF0C9U 86263251 IC50 = 321 nM T25637 C5U0ZG 117949685 IC50 = 2511.89 nM T25637 CCG05U 117949686 IC50 = 316.23 nM T25637 C3UBY0 122163387 IC50 = 310 nM T25637 C4P9JW 122516179 IC50 = 370 nM T25637 CYT3P6 122516185 IC50 = 2900 nM T25637 CMB23H 122516211 IC50 = 62 nM T25637 CV25IT 122516222 IC50 = 110 nM T25637 CU9N2M 122516246 IC50 = 270 nM T25637 CN3VC8 122516255 IC50 = 53 nM T25637 C4M3ZK 122516295 IC50 = 56 nM T25637 C4ELG0 122516336 IC50 = 50 nM T25637 C9BL6C 122516346 IC50 = 500 nM T25637 CX3B4R 122516830 IC50 = 140 nM T25637 C41DZW 122516838 IC50 = 67 nM T25637 COK0J3 122516959 IC50 = 62 nM T25637 C0AQW4 122517020 IC50 = 570 nM T25637 CL3Q9Z 122517043 IC50 = 130 nM T25637 CCAF42 130302575 IC50 = 50.12 nM T25637 C2QC4N 130302611 IC50 = 25.12 nM T25637 C84UJE 130302628 IC50 = 13 nM T25637 C73YSW 130302637 IC50 = 794.33 nM T25637 CY4E5Q 130302665 IC50 = 125.89 nM T25637 C2UIN3 130302696 IC50 = 19.95 nM T25637 CY50ZM 130302793 IC50 = 125.89 nM T25637 C7J8OU 130344903 IC50 = 255 nM T25637 CK1G8Z 130344958 IC50 = 671 nM T25637 C4NT5Q 130344969 IC50 = 174 nM T25637 C3M2IV 130344977 IC50 = 103 nM T25637 C5H6ZM 130345003 IC50 = 310 nM T25637 CE8Q7I 130345035 IC50 = 126 nM T25637 C01UGK 130345060 IC50 = 380 nM T25637 CN9S7B 130345097 IC50 = 120 nM T25637 C3CH7B 130345110 IC50 = 78 nM T25637 CC10LU 130345138 IC50 = 259 nM T25637 C0VMZ6 130345145 IC50 = 423 nM T25637 CW53BD 130345152 IC50 = 192 nM T25637 C7RN8L 130345158 IC50 = 2200 nM T25637 C3DS1X 130345159 IC50 = 686 nM T25637 CF20BS 130345178 IC50 = 69 nM T25637 CB0YI5 130345191 IC50 = 470 nM T25637 CMO50A 130345200 IC50 = 2000 nM T25637 CY04NF 130345225 IC50 = 606 nM T25637 CA9QM5 130345306 IC50 = 343 nM T25637 CSRB12 130345397 IC50 = 1040 nM T25637 C3BHA0 130358066 IC50 = 342 nM T25637 C7M2GA 130358093 IC50 = 2164 nM T25637 CLSP06 130358333 IC50 = 828 nM T25637 C29WVS 130358344 IC50 = 176 nM T25637 CZM13E 130358354 IC50 = 143 nM T25637 C40NJZ 130358433 IC50 = 397 nM T25637 CL74FP 132253032 IC50 = 110 nM T25637 CSEW98 132253084 IC50 = 78 nM T25637 CG6KP2 132253106 IC50 = 58 nM T25637 CCL91Y 132253144 IC50 = 35 nM T25637 C4C6HK 132253151 IC50 = 77 nM T25637 CJAN-32 132253163 IC50 = 43 nM T25637 CC89LI 132253175 IC50 = 9900 nM T25637 CS0LC7 134280641 IC50 = 81 nM T25637 CGN6E7 135492608 IC50 = 1000 nM T25637 CC35GR 135615984 IC50 = 34000 nM T25637 C93RLN 137459807 IC50 = 3162.28 nM T25637 CX83CB 137459827 IC50 = 5.012 nM T25637 CI8C3G 137459832 IC50 = 79.43 nM T25637 CAK9N2 137459833 IC50 = 63.1 nM T25637 C9P4YE 137459864 IC50 = 100 nM T25637 CE9O8V 137634616 IC50 = 74 nM T25637 C7DIT4 137645206 IC50 > 31000 nM T25637 CI1Y2F 137648233 IC50 = 180 nM T25637 CTA4O6 137656044 IC50 = 82 nM T25637 C1JKW0 138648299 IC50 = 3190 nM T25637 C6F3IB 140959818 IC50 = 501.19 nM T25637 C3WV9D 140959830 IC50 = 79.43 nM T25637 C74QLH 145712358 IC50 = 19.95 nM T25637 CR62OV 155515216 IC50 = 316.23 nM T25637 CUL8C7 155515256 IC50 = 233 nM T25637 C86LXI 155515261 IC50 = 236 nM T25637 CC6NO1 155516293 IC50 = 794.33 nM T25637 C9X0ZG 155522519 IC50 = 199.53 nM T25637 CI0V5F 155525579 IC50 = 69 nM T25637 CG4CH3 155527512 IC50 = 794.33 nM T25637 CG38CQ 155527837 IC50 = 68260 nM T25637 CABH27 155529596 IC50 = 100 nM T25637 CQV98K 155531889 IC50 = 19.95 nM T25637 CZ4Y7A 155532323 IC50 = 554 nM T25637 CP35IW 155532402 IC50 = 184 nM T25637 CS2OJ7 155533774 IC50 = 1995.26 nM T25637 CCN0P3 155545992 IC50 = 19.95 nM T25637 CC36QH 155546157 IC50 = 251.19 nM T25637 C8RS5F 155549747 IC50 = 394 nM T25637 CWL16Z 155550534 IC50 = 85 nM T25637 CEW2G4 155555668 IC50 = 652 nM T25637 CI56NY 155555837 IC50 = 794.33 nM T25637 CEHP09 155556842 IC50 = 12.59 nM T25637 CFS17Y 155557978 IC50 = 1596 nM T25637 C0AU7O 155560147 IC50 = 280 nM T25637 CA35OS 155560404 IC50 = 50.12 nM T25637 CH93UL 155561434 IC50 = 125.89 nM T25637 COF96P 155564105 IC50 = 146 nM T25637 CKLG01 155567035 IC50 = 794.33 nM T25637 D02UVS 5455 IC50 = 170 nM T25637 D0Q6PI 1001 IC50 = 60100 nM T87020 D0G7UX 5284373 IC50 = 16 nM T87020 D02VJY 3037617 IC50 = 7370 nM T87020 D04PGB 445501 IC50 > 100000 nM T87020 C1RN6G 445646 Ki = 100000 nM T87020 C4DR9Q 3350117 Ki = 290000 nM T87020 C2HUW7 5282071 IC50 = 8000 nM T87020 C6W4CX 5496888 IC50 = 540000 nM T87020 C1I0LW 6540258 IC50 = 1450000 nM T87020 CRD1T0 9811664 IC50 > 100000 nM T87020 C9IS6O 9820942 IC50 > 150000 nM T87020 C5S6IB 9822783 Ki = 90000 nM T87020 CSN72K 10371065 IC50 = 9370 nM T87020 CF3GI4 10508532 Ki > 500000 nM T87020 CJ10LB 10628798 IC50 = 325000 nM T87020 CAC94N 10700607 IC50 = 365000 nM T87020 C5NB9Z 11129344 IC50 > 100000 nM T87020 CTLC58 35027274 IC50 = 1070 nM T87020 CA8G7V 44294786 IC50 > 10000000 nM T87020 C5KU2V 44339314 Ki = 190000 nM T87020 CR93AH 44339414 Ki = 340000 nM T87020 C5A8UB 44339420 Ki = 11000000 nM T87020 CKDT15 44339421 Ki = 2900000 nM T87020 C0WA3X 44339433 Ki = 840000 nM T87020 CFL1Y9 44350840 IC50 = 215000 nM T87020 CFSE98 44350865 IC50 = 15000 nM T87020 CTH57E 44387378 IC50 = 28000 nM T87020 C2V6RJ 56962328 IC50 = 4200 nM T87020 CJ46RD 56962330 IC50 = 3500 nM T87020 C1BUW4 57521458 IC50 = 6200 nM T87020 CGU89M 57521460 IC50 > 100000 nM T87020 CKP31Q 57521461 IC50 = 2800 nM T87020 C7D3PN 57521557 IC50 = 5550 nM T87020 CO6T0F 57521558 IC50 = 11600 nM T87020 C2RVN0 57521777 IC50 = 2130 nM T87020 C8PY2R 57521778 IC50 = 2880 nM T87020 C0HOD9 57521879 IC50 = 2200 nM T87020 CS7B2A 57521880 IC50 = 2640 nM T87020 CGP03D 57521881 IC50 > 100000 nM T87020 C9V4QB 57521882 IC50 = 32800 nM T87020 C4C7LK 57522005 IC50 = 32500 nM T87020 C8YI0U 57522006 IC50 > 100000 nM T87020 C0KC6J 57522007 IC50 > 100000 nM T87020 CH89PN 57522008 IC50 = 69900 nM T87020 CG6TK3 57522120 IC50 > 100000 nM T87020 CWQ8J7 57522121 IC50 > 100000 nM T87020 CTCH51 57522237 IC50 = 84500 nM T87020 C8R2IJ 57522238 IC50 = 15690 nM T87020 C1PBX3 57522239 IC50 = 14300 nM T87020 CU5NP7 57522240 IC50 > 100000 nM T87020 C0P3TI 57522347 IC50 > 100000 nM T87020 C6WY9D 57522348 IC50 = 40300 nM T87020 C6FQ4X 57522350 IC50 > 100000 nM T87020 CHVK79 57522455 IC50 > 100000 nM T87020 C73XQS 57522456 IC50 > 100000 nM T87020 C4OJX2 57522457 IC50 = 20300 nM T87020 CGIX69 57522458 IC50 = 17700 nM T87020 CG2SO6 57522567 IC50 = 20500 nM T87020 CR9C3F 57522569 IC50 = 43900 nM T87020 C8SP3L 57522570 IC50 > 100000 nM T87020 CQ3I7G 57522682 IC50 = 26500 nM T87020 C5QM2O 57522683 IC50 = 66500 nM T87020 CE7G2U 57522684 IC50 > 100000 nM T87020 CA4R9I 57522685 IC50 > 100000 nM T87020 C3EP9M 57522800 IC50 > 100000 nM T87020 C46EIF 57522801 IC50 > 100000 nM T87020 CC85GJ 57522802 IC50 > 50000 nM T87020 CCUW31 57522803 IC50 > 50000 nM T87020 CV58SP 57522927 IC50 = 41600 nM T87020 CT58KB 57522928 IC50 = 710 nM T87020 C95OGY 57522929 IC50 > 50000 nM T87020 CZI07G 57522930 IC50 = 3410 nM T87020 C8B9HE 57522931 IC50 = 8300 nM T87020 C7Y9SK 57523063 IC50 = 49200 nM T87020 C4S5KW 57523064 IC50 > 100000 nM T87020 CT4NB0 57523068 IC50 > 100000 nM T87020 C0NUH8 57523069 IC50 > 100000 nM T87020 C2YN0S 57523070 IC50 = 15130 nM T87020 C7BR2S 59925440 Ki = 30000 nM T87020 C2DIM5 70684253 IC50 > 100000 nM T87020 CYQH64 70684260 IC50 = 3720 nM T87020 CG5D2W 70688508 IC50 > 100000 nM T87020 CWDU09 70688522 IC50 = 9770 nM T87020 CWY7C0 70692710 IC50 = 11700 nM T87020 C5MK3W 70694725 IC50 > 100000 nM T87020 CD65LN 70694726 IC50 > 100000 nM T87020 CEZG14 70694756 IC50 > 100000 nM T87020 CU9RN3 70694757 IC50 = 890 nM T87020 CJ2H0K 73353060 IC50 = 640000 nM T87020 C5EMH2 86277875 Ki > 50000 nM T87020 CWTL26 117967814 Ki > 500000 nM T87020 CTI1X7 117968005 Ki > 1000000 nM T87020 CNP23H 122192627 Ki > 50000 nM T87020 CEMN03 122192628 Ki > 100000 nM T87020 C5ZF3W 122192629 Ki = 9700 nM T87020 C1P6LO 137642835 Ki = 18.9 nM T87020 D06ZWX 6197 Ki = 24200 nM T81735 D09XZB 123631 IC50 > 50000 nM T81735 D0B3HD 2519 IC50 = 10000000 nM T81735 D0E6XR 3062316 IC50 > 50000 nM T81735 D0J5VR 11625818 IC50 = 6700 nM T81735 D0R0MW 5329102 IC50 > 50000 nM T81735 D0R4OM 5566 IC50 = 100000 nM T81735 D0W5HK 216239 IC50 > 50000 nM T81735 D01QSO 16654980 IC50 = 6917 nM T81735 D06DMQ 59472121 Ki > 4000 nM T81735 D08OOJ 73051434 IC50 = 500 nM T81735 D08QGT 17755052 IC50 = 1230 nM T81735 D0H2UB 5361 IC50 = 1700 nM T81735 D0H9DA 54761306 IC50 > 30000 nM T81735 D0I3LO 91933883 IC50 = 4800 nM T81735 D0O1IM 58298318 IC50 = 15 nM T81735 D0TU7B 58507717 IC50 = 8567 nM T81735 D0UP1Z 51001932 IC50 > 4800 nM T81735 D0W7HE 56649450 IC50 > 9100 nM T81735 D0XD4I 118502708 IC50 = 140 nM T81735 D03BNU 59604787 IC50 = 8831 nM T81735 D0B5YS 1183 IC50 = 1500000 nM T81735 D05HIJ 135565159 IC50 = 2000 nM T81735 D09SFV 3973 IC50 = 300 nM T81735 D0P1JI 312145 Ki = 120 nM T81735 CBSY87 79351 IC50 = 30000 nM T81735 C51ZJH 88505 IC50 = 15000 nM T81735 CAUK86 108130 IC50 > 1000000000 nM T81735 CN41ZV 2834824 IC50 > 10000 nM T81735 CE74CV 5059890 IC50 = 420 nM T81735 CE1Y8A 9815659 IC50 = 400 nM T81735 C93ZDI 9817915 IC50 = 280 nM T81735 CGR32P 9835264 IC50 = 530 nM T81735 CK41WR 9843885 IC50 = 160 nM T81735 C0V4QC 9994599 IC50 > 10000 nM T81735 CI15ET 10074436 IC50 = 130 nM T81735 CE0N7T 10470014 IC50 = 35 nM T81735 CC79PE 10708932 IC50 > 10000 nM T81735 C2QWF1 10802700 IC50 > 10000 nM T81735 C60WVN 11162233 IC50 > 10000 nM T81735 CEP34D 11175067 IC50 > 10000 nM T81735 CL21AE 11184764 IC50 > 10000 nM T81735 CF0RP8 11185299 IC50 > 10000 nM T81735 CQN95X 11185524 IC50 > 10000 nM T81735 C0YI4E 11220585 IC50 > 10000 nM T81735 CL8YE3 11230964 IC50 = 250 nM T81735 CZG5F0 11232354 IC50 > 10000 nM T81735 C2I8TN 11243737 IC50 > 10000 nM T81735 C91YKC 11255019 IC50 > 10000 nM T81735 CL6M9W 11256465 IC50 > 10000 nM T81735 C6QOP3 11256466 IC50 = 10470 nM T81735 COHR75 11266772 IC50 > 10000 nM T81735 CVJ4N2 11278356 IC50 > 10000 nM T81735 CUH49V 11281305 IC50 > 10000 nM T81735 C97UDS 11312053 IC50 = 9270 nM T81735 C4SKU3 11322952 IC50 > 10000 nM T81735 C5QES9 11323606 IC50 = 8460 nM T81735 C9YM3B 11336414 IC50 > 10000 nM T81735 CM4TV0 11346543 IC50 = 6490 nM T81735 CBEJ76 11347335 IC50 > 10000 nM T81735 C4O8WG 11347336 IC50 > 10000 nM T81735 C78AXV 11359006 IC50 > 10000 nM T81735 CRSY04 11359736 IC50 = 5710 nM T81735 CWC89E 11369108 IC50 = 6680 nM T81735 CQ9T0H 11370302 IC50 = 6710 nM T81735 CIO3M7 11381536 IC50 > 10000 nM T81735 CJ3LG8 11392135 IC50 > 10000 nM T81735 C5QX9B 11393330 IC50 > 10000 nM T81735 C4CZ5K 11402810 IC50 = 2810 nM T81735 CT12HC 11414529 IC50 > 10000 nM T81735 C0MIO7 11415324 IC50 > 10000 nM T81735 CWT7D5 11437813 IC50 = 3190 nM T81735 CK0WT9 11439424 IC50 > 10000 nM T81735 CJGL73 11470834 IC50 > 10000 nM T81735 C9QFU2 11471412 IC50 > 10000 nM T81735 CR6QP2 11494112 IC50 = 8180 nM T81735 C03LVG 11507468 IC50 > 10000 nM T81735 CEM84I 11508579 IC50 = 3940 nM T81735 CN70WA 11508681 IC50 = 800 nM T81735 CL36GP 11516053 IC50 = 4000 nM T81735 CL6MF0 11516928 IC50 = 2300 nM T81735 C2UN5J 11517255 IC50 = 560 nM T81735 CY47AQ 11519784 EC50 = 426 nM T81735 C1PYA4 11521848 IC50 > 10000 nM T81735 CC5V8Q 11523982 IC50 > 30000 nM T81735 CXH0E7 11524058 IC50 = 3940 nM T81735 C0YHE4 11527442 IC50 = 7 nM T81735 CWFC48 11529127 IC50 > 10000 nM T81735 CC4WA6 11530666 IC50 = 14700 nM T81735 CX8RW9 11532281 IC50 = 3500 nM T81735 C7WK9H 11536329 IC50 > 10000 nM T81735 C1VA4C 11543481 IC50 = 150 nM T81735 C8H2MI 11544508 IC50 = 4900 nM T81735 CH0X7Y 11544698 IC50 = 940 nM T81735 C15EOX 11545136 IC50 = 8900 nM T81735 C76DGX 11545472 IC50 > 10000 nM T81735 CDI1G8 11550883 IC50 > 10000 nM T81735 CL12DP 11552413 IC50 > 10000 nM T81735 CHV4F5 11552464 IC50 = 8700 nM T81735 CBZ6E1 11552974 IC50 = 840 nM T81735 CA59NY 11553441 IC50 = 470 nM T81735 CV2UO9 11554515 IC50 = 9700 nM T81735 CO9H6K 11558264 IC50 > 10000 nM T81735 CACS26 11561968 Ki > 10000 nM T81735 CS0OL9 11567907 IC50 = 23 nM T81735 CQZC21 11574915 IC50 = 8490 nM T81735 CZO4A7 11575363 IC50 = 4330 nM T81735 C2EB5G 11580379 IC50 = 530 nM T81735 CNI7P8 11581520 IC50 = 500 nM T81735 CZH7G2 11584859 IC50 = 11 nM T81735 C2L1AP 11585185 IC50 = 30 nM T81735 CW64QL 11588083 IC50 = 2900 nM T81735 CZ7PA3 11588581 IC50 = 690 nM T81735 C0MEC7 11588610 IC50 = 800 nM T81735 C8WT0U 11589142 IC50 = 440 nM T81735 CZA43X 11594202 IC50 = 10000 nM T81735 C69LMH 11594375 IC50 > 10000 nM T81735 CBJ08E 11594997 IC50 > 10000 nM T81735 CAK3G2 11595733 IC50 > 30000 nM T81735 CE3RC2 11595862 IC50 = 490 nM T81735 CJGV32 11602760 IC50 = 800 nM T81735 CO3A8B 11603526 IC50 = 1400 nM T81735 CV8W7G 11604008 IC50 > 10000 nM T81735 C31IBM 11610438 IC50 = 2530 nM T81735 C5MWL6 11610829 IC50 > 30000 nM T81735 CM10KH 11611160 IC50 = 4300 nM T81735 CBH6F5 11616783 IC50 > 10000 nM T81735 CX3Y6B 11628492 IC50 = 4 nM T81735 CW08IG 11631748 IC50 = 440 nM T81735 CN0UG9 11633358 IC50 = 4130 nM T81735 CG86TF 11633621 IC50 > 30000 nM T81735 C2LV9M 11637988 IC50 > 10000 nM T81735 CTBU41 11638873 IC50 = 1100 nM T81735 CR5K4P 11640310 IC50 = 8150 nM T81735 C5B7LF 11642233 IC50 = 16 nM T81735 CGR73T 11645742 IC50 = 4000 nM T81735 C81TOS 11652482 IC50 > 10000 nM T81735 CK85WO 11653341 IC50 > 30000 nM T81735 C38OLX 11653621 IC50 = 790 nM T81735 CU3RW5 11654534 IC50 = 26600 nM T81735 C8WP6A 11659962 IC50 > 10000 nM T81735 C0Z2LD 11660078 IC50 = 600 nM T81735 C8LA7J 11660443 IC50 > 30000 nM T81735 CP67TA 11660662 IC50 > 10000 nM T81735 COE5R0 11675561 IC50 = 9440 nM T81735 C67IHX 11676414 IC50 = 350 nM T81735 C91EYU 11678629 IC50 = 6 nM T81735 CZJE78 11681727 IC50 > 10000 nM T81735 CKR62Z 11681912 IC50 = 3000 nM T81735 CQM40U 11682080 IC50 > 30000 nM T81735 CKMD57 11683057 IC50 = 5900 nM T81735 CQZ42E 11688386 IC50 = 34 nM T81735 CS7ZN2 11688948 IC50 > 10000 nM T81735 CKPC75 11689114 IC50 = 1200 nM T81735 CH9K8U 11689409 IC50 = 2700 nM T81735 CU0E8O 11690457 Ki > 10000 nM T81735 C4F9CK 11692871 IC50 = 7 nM T81735 C78MCL 11694511 IC50 > 10000 nM T81735 CR8OX0 11696073 IC50 = 9320 nM T81735 C0OR1Y 11696317 IC50 = 3760 nM T81735 C4QFH8 11696624 IC50 > 10000 nM T81735 CYKE69 11697295 IC50 = 2000 nM T81735 CD61KM 11701732 IC50 > 10000 nM T81735 C8VX5H 11703673 IC50 = 710 nM T81735 CCVY97 11704378 IC50 = 1920 nM T81735 CB0AP2 11705863 Ki > 10000 nM T81735 CO81SN 11709138 IC50 > 10000 nM T81735 C0K5MT 11711208 IC50 > 10000 nM T81735 CZ07SN 11717521 IC50 = 3100 nM T81735 CE37NP 11717869 IC50 = 3100 nM T81735 CO5A2S 11718914 IC50 = 5580 nM T81735 CBC3Z9 11721120 IC50 = 14 nM T81735 CQ1JW7 11721214 IC50 = 55 nM T81735 CU87RX 11721385 IC50 = 38 nM T81735 C8QE5A 11737711 IC50 = 360 nM T81735 C4PGI6 11737755 IC50 > 10000 nM T81735 C4EX0L 11738398 IC50 = 3520 nM T81735 C4N1LD 11771277 IC50 = 3250 nM T81735 C1N4TD 11956265 IC50 = 510 nM T81735 C9MF8V 11956267 IC50 = 3010 nM T81735 C4LV1C 11956268 IC50 = 1070 nM T81735 CCP9B7 11956322 IC50 = 490 nM T81735 C9EOB2 11956323 IC50 = 360 nM T81735 CC45GI 11956324 IC50 = 640 nM T81735 C2US9R 12341861 IC50 > 10000 nM T81735 CX9I4D 12896644 IC50 = 6500 nM T81735 C1SNR6 13141222 IC50 > 8000 nM T81735 CY7A0T 14638904 IC50 = 1600 nM T81735 C56LPQ 15950788 IC50 = 13 nM T81735 CPY21E 16203245 IC50 = 160 nM T81735 C4MJ9Z 16203247 IC50 = 260 nM T81735 C2AXJ7 16203250 IC50 = 6300 nM T81735 CAI9S5 16203254 IC50 = 1300 nM T81735 C1I8YQ 16203357 IC50 = 4200 nM T81735 CGQ82D 16203358 IC50 = 1800 nM T81735 C9E4OH 16203360 IC50 = 1000 nM T81735 C42FYM 16203361 IC50 = 8800 nM T81735 C0BM7J 16203362 IC50 = 920 nM T81735 CY9GT0 16203364 IC50 = 350 nM T81735 CGVM24 16203466 IC50 > 100000 nM T81735 CN7QP8 16203467 IC50 = 1300 nM T81735 C5KUF9 16203476 IC50 = 680 nM T81735 C4WI3R 16203581 IC50 > 100000 nM T81735 C73CJI 16203583 IC50 > 10000 nM T81735 CR2S5J 16203591 IC50 = 19000 nM T81735 CD4XG7 16203592 IC50 = 15000 nM T81735 C3FWM9 16203595 IC50 = 1000 nM T81735 CGO9N1 16203602 IC50 = 3600 nM T81735 CY1EH7 16203710 IC50 > 100000 nM T81735 CGD2B4 16203711 IC50 > 100000 nM T81735 CFN79L 16203713 IC50 = 700 nM T81735 CED0M3 16203716 IC50 = 11000 nM T81735 C79JLP 16203721 IC50 = 3600 nM T81735 CK2Q7B 16203821 IC50 = 920 nM T81735 C0RO4Y 16203822 IC50 > 30000 nM T81735 CLJT07 16203823 IC50 > 100000 nM T81735 CW2X8R 16203825 IC50 > 100000 nM T81735 C34PTV 16203827 IC50 > 100000 nM T81735 CZ9V3G 16203828 IC50 > 100000 nM T81735 C5J7FQ 16203836 IC50 = 1100 nM T81735 C2JA8F 16203837 IC50 = 3200 nM T81735 CQ1Z0V 16203940 IC50 = 500 nM T81735 C45LZB 16203944 IC50 = 4200 nM T81735 C4SJX6 16203947 IC50 = 3600 nM T81735 C7TOJ8 16203948 IC50 = 600 nM T81735 CODI71 16204048 IC50 = 9700 nM T81735 CNCV97 16204163 IC50 > 100000 nM T81735 C91SAQ 16204164 IC50 > 100000 nM T81735 C1G6DV 16204249 IC50 = 680 nM T81735 CF1ET3 16204250 IC50 = 2100 nM T81735 C47PLJ 16204251 IC50 = 1900 nM T81735 C6W7LV 16204252 IC50 = 7300 nM T81735 C08QGM 16204253 IC50 > 100000 nM T81735 C48POT 16204254 IC50 > 100000 nM T81735 C4C3QB 16204255 IC50 > 100000 nM T81735 CZ7DW6 16204460 IC50 = 840 nM T81735 CV9US5 16736978 IC50 > 10000 nM T81735 CF6JS9 16757570 IC50 = 1500 nM T81735 C1SN9M 17756679 IC50 = 500 nM T81735 CV6P2N 19088789 IC50 = 910 nM T81735 CQ4ZT1 21106427 IC50 = 3200 nM T81735 C7N8CH 21106429 IC50 = 390 nM T81735 CT5G7O 21955998 IC50 = 480 nM T81735 CP05ZB 22346757 IC50 = 5000 nM T81735 C1F2TM 23582995 IC50 = 300 nM T81735 C2GK1J 23583257 IC50 = 6800 nM T81735 CEYL29 23585510 IC50 > 10000 nM T81735 CBL37C 23642173 IC50 > 10000 nM T81735 CM9C0R 24866805 IC50 = 780 nM T81735 CB79YC 24905143 IC50 = 190 nM T81735 C2DC9J 24905144 IC50 = 29 nM T81735 CN6V8Z 24905145 IC50 = 17 nM T81735 CSB7P5 24905148 IC50 = 53 nM T81735 CGSF21 24905149 IC50 = 48000 nM T81735 CVDG02 24905150 IC50 = 6400 nM T81735 CWH6C5 24905152 IC50 = 8 nM T81735 C0HE2Q 24905153 IC50 = 47 nM T81735 C7QSC9 24905154 IC50 = 339 nM T81735 CO9D0K 24905155 IC50 = 1960 nM T81735 C5W9UR 24905157 IC50 = 184 nM T81735 CC1DA3 24905158 IC50 = 737 nM T81735 COW79F 24905159 IC50 = 365 nM T81735 CFPA53 24905160 IC50 = 1230 nM T81735 C2O0JX 24905161 IC50 = 979 nM T81735 CA72BE 24905162 IC50 = 713 nM T81735 CQN6X9 24905163 IC50 = 288 nM T81735 CD4O1F 24905165 IC50 = 1200 nM T81735 CKL48T 24905166 IC50 = 2680 nM T81735 C76VYL 24905167 IC50 = 883 nM T81735 C7K5PU 24905168 IC50 = 331 nM T81735 CZ57ID 24905169 IC50 = 1260 nM T81735 C2DHX9 24905170 IC50 = 2750 nM T81735 CSB96E 24905171 IC50 = 10100 nM T81735 CWZ0R2 24905172 IC50 = 489 nM T81735 CY3B6M 24905175 IC50 = 824 nM T81735 CW7UA3 24905176 IC50 = 873 nM T81735 CW1V0H 24905177 IC50 = 3410 nM T81735 CO6Y0L 24905178 IC50 = 2270 nM T81735 C60NQW 24905179 IC50 = 789 nM T81735 C4MO8B 24905180 IC50 = 251 nM T81735 COJI47 24905181 IC50 = 185 nM T81735 CS0B2C 24905182 IC50 = 919 nM T81735 C1H4BT 24905183 IC50 = 509 nM T81735 C4WHK9 24905184 IC50 = 826 nM T81735 C7Q4MZ 24905185 IC50 = 430 nM T81735 CS4IP1 24905186 IC50 = 309 nM T81735 C69QWO 24905187 IC50 = 916 nM T81735 C85ANB 24905188 IC50 = 90 nM T81735 CNHD75 24905189 IC50 = 463 nM T81735 C9JUO2 24905190 IC50 = 953 nM T81735 CPR03K 24905191 IC50 = 929 nM T81735 CTAG19 24905193 IC50 = 80 nM T81735 C7VJM5 24905194 IC50 = 546 nM T81735 CEP1L3 24905195 IC50 = 303 nM T81735 CP68ZD 24905196 IC50 = 220 nM T81735 C8Z0RJ 24905197 IC50 = 383 nM T81735 CN9RT0 24905198 IC50 = 5800 nM T81735 CHI78P 24905200 IC50 = 317 nM T81735 CO6PE8 24905201 IC50 = 88 nM T81735 CZ63HS 24905202 IC50 = 71 nM T81735 C2X0FC 24905203 IC50 = 77 nM T81735 C0WCE3 24905204 IC50 = 36 nM T81735 CNK50B 24905205 IC50 = 47 nM T81735 C12DPB 24905206 IC50 = 110 nM T81735 C8N0RH 24905207 IC50 = 260 nM T81735 CYA5G2 24905208 IC50 = 102 nM T81735 CDV2B4 24905209 IC50 = 150 nM T81735 CEFK68 24905210 IC50 = 120 nM T81735 CUFP12 24905211 IC50 = 214 nM T81735 C0JG8L 24905212 IC50 = 54 nM T81735 CP47MK 24905213 IC50 = 5000 nM T81735 CB61QC 24905214 IC50 = 5000 nM T81735 CQ13ZI 24905215 IC50 = 2700 nM T81735 C6VI8F 24905216 IC50 = 80 nM T81735 CXNH25 24905217 IC50 = 49 nM T81735 C2PN9S 24905218 IC50 = 126 nM T81735 C9O2AL 24905219 IC50 = 359 nM T81735 CIT7U8 24905220 IC50 = 1100 nM T81735 CMD26S 24905221 IC50 = 349 nM T81735 C4R8WC 24905222 IC50 = 244 nM T81735 C47SHA 24905223 IC50 = 105 nM T81735 C1DY2R 24905224 IC50 = 85 nM T81735 CS0XF9 24905225 IC50 = 8100 nM T81735 CG5VX2 24905226 IC50 = 18000 nM T81735 C57QEO 24905227 IC50 = 100000 nM T81735 C7CG5E 24905228 IC50 = 314 nM T81735 CHP5D1 24905229 IC50 = 260 nM T81735 CXP09S 24905230 IC50 = 46 nM T81735 CY7XG1 24905231 IC50 = 1900 nM T81735 C7JFQ2 24905232 IC50 = 14 nM T81735 C2JM1P 24905233 IC50 = 2000 nM T81735 CC3BF0 24905234 IC50 = 283 nM T81735 CE57FI 24905235 IC50 = 100000 nM T81735 CUP20O 24905236 IC50 = 6000 nM T81735 CLC6Q2 24905237 IC50 = 2600 nM T81735 C9M1GI 24905238 IC50 = 216 nM T81735 CVD72F 24905239 IC50 = 10 nM T81735 CK38IZ 24905240 IC50 = 9 nM T81735 CO2V5E 24905241 IC50 = 186 nM T81735 CZBA19 24905244 IC50 = 3400 nM T81735 CQ8OI1 24905246 IC50 = 222 nM T81735 C5URC6 24905247 IC50 = 400 nM T81735 CZ2E9K 24905249 IC50 = 280 nM T81735 C03SVO 24905250 IC50 = 1300 nM T81735 CIF2J5 24905251 IC50 = 640 nM T81735 CPTE58 24905252 IC50 = 717 nM T81735 CX1JB8 24905253 IC50 = 1100 nM T81735 COZ3H7 24905254 IC50 = 7100 nM T81735 CDT1H9 24905255 IC50 = 3700 nM T81735 C54QKA 24905256 IC50 = 440 nM T81735 C9U0JA 24905259 IC50 = 400 nM T81735 CO4YS7 24905260 IC50 = 2400 nM T81735 CEG0B5 24905261 IC50 = 100000 nM T81735 C9VE5F 24905262 IC50 = 100000 nM T81735 C3I4HK 24905264 IC50 = 670 nM T81735 C0VMI6 24905265 IC50 = 100000 nM T81735 CWE3V0 24905267 IC50 = 100000 nM T81735 CH4T3A 24905268 IC50 = 4400 nM T81735 CVT17Q 24905270 IC50 = 210 nM T81735 C6QDN7 24905271 IC50 = 350 nM T81735 C6XHJ7 24905272 IC50 = 200 nM T81735 CTB9A3 24905273 IC50 = 2100 nM T81735 C0NB1Q 24905274 IC50 = 340 nM T81735 C9KQ0L 24905275 IC50 = 630 nM T81735 C9O8QZ 24905277 IC50 = 880 nM T81735 CP50RD 24905280 IC50 = 88 nM T81735 CG13ZM 24905281 IC50 = 100000 nM T81735 CF0S6X 24905282 IC50 = 847 nM T81735 C5HBL0 24905284 IC50 = 24300 nM T81735 C2Z5DN 24905285 IC50 = 478 nM T81735 CL6GH8 24905286 IC50 = 576 nM T81735 CKYO98 24905287 IC50 = 212 nM T81735 CRNQ65 24905288 IC50 = 212 nM T81735 COD7I5 24905289 IC50 = 336 nM T81735 C4LP7E 24905290 IC50 = 173 nM T81735 CE9JC2 24905291 IC50 = 150 nM T81735 C2GI1R 24905292 IC50 = 2020 nM T81735 CHW8C4 24905293 IC50 = 214 nM T81735 CQF0H1 24905294 IC50 = 111 nM T81735 CNO7X0 24905295 IC50 = 17 nM T81735 C5WRG7 24905296 IC50 = 242 nM T81735 CQ1S0U 24905297 IC50 = 556 nM T81735 C4UES7 24905298 IC50 = 2500 nM T81735 CMS69P 24905299 IC50 = 1930 nM T81735 CC0U5M 24905300 IC50 = 13 nM T81735 CW7X6S 24905301 IC50 = 2740 nM T81735 C97IQV 24905302 IC50 = 110 nM T81735 CSJ47V 24905303 IC50 = 408 nM T81735 CPN74C 24905304 IC50 = 367 nM T81735 C5CS3N 24905305 IC50 = 169 nM T81735 CK4XE9 24905307 IC50 = 49 nM T81735 CTU6Z3 24905308 IC50 = 3690 nM T81735 C9SQX1 24905309 IC50 = 543 nM T81735 CM75JP 24905310 IC50 = 610 nM T81735 C9Q2BJ 24905311 IC50 = 1310 nM T81735 C9VUA1 24905312 IC50 = 77 nM T81735 CU3RS1 24905313 IC50 = 683 nM T81735 CYG3H2 24905314 IC50 = 242 nM T81735 CV5Q7O 24905315 IC50 = 107 nM T81735 C8SA3O 24905316 IC50 = 155 nM T81735 CI5MN3 24905317 IC50 = 28 nM T81735 CJ1P7K 24905318 IC50 = 35 nM T81735 C1T6YQ 24905319 IC50 = 151 nM T81735 CAU86X 24905320 IC50 = 277 nM T81735 C54ISY 24905321 IC50 = 1610 nM T81735 C2GE5I 24905322 IC50 = 180 nM T81735 C8D6YK 24905323 IC50 = 500 nM T81735 C5NZH9 24905324 IC50 = 64 nM T81735 C9D6JR 24905325 IC50 = 336 nM T81735 CLZT41 24905326 IC50 = 43 nM T81735 CW8FD3 24905327 IC50 = 370 nM T81735 CHB7A2 24905328 IC50 = 194 nM T81735 CA8EI3 24905329 IC50 = 149 nM T81735 CCQ0O7 24905330 IC50 = 1300 nM T81735 CJ81AS 24905331 IC50 = 12 nM T81735 C8PW4H 24905332 IC50 = 19 nM T81735 C2Y5TF 24905333 IC50 = 30 nM T81735 CH9FL5 24905334 IC50 = 660 nM T81735 C1S0PC 24905335 IC50 = 709 nM T81735 C8N9MV 24905336 IC50 = 218 nM T81735 C9E8BJ 24905338 IC50 = 894 nM T81735 CX85AC 24905341 IC50 = 4280 nM T81735 CKZ80E 24905342 IC50 = 735 nM T81735 CO8SH1 24905343 IC50 = 439 nM T81735 C7IZL6 24905344 IC50 = 1350 nM T81735 C78UAX 25169571 IC50 = 8 nM T81735 CA3B6H 25169574 IC50 = 12 nM T81735 CBM07Q 25169777 IC50 = 51 nM T81735 CYU48A 25169778 IC50 = 2 nM T81735 CFEW09 25169995 IC50 = 10 nM T81735 CV9WY2 25169996 IC50 = 21 nM T81735 CX7WQ8 25169999 IC50 = 8 nM T81735 CNQB64 25170200 IC50 = 8 nM T81735 CJ0DW4 25170201 IC50 = 9 nM T81735 CIQ2O1 25170593 IC50 = 6 nM T81735 C05QSJ 25170594 IC50 = 7 nM T81735 C7C0IY 25170783 IC50 = 2 nM T81735 CMV9H2 25171023 IC50 = 41 nM T81735 CTO1K8 25171024 IC50 = 7 nM T81735 CM93HP 25172264 IC50 = 6 nM T81735 C5TJD2 25172265 EC50 = 109 nM T81735 CDA4L9 25172657 IC50 = 3 nM T81735 CQG02I 25211673 IC50 = 18 nM T81735 C4KX1S 44328172 IC50 > 500000 nM T81735 CSHJ14 44383813 IC50 = 20 nM T81735 C5N2CH 44388148 IC50 = 4140 nM T81735 CJ4I2B 44397050 IC50 = 900 nM T81735 C8X1UZ 44405259 IC50 = 6200 nM T81735 CWYN01 44405265 IC50 = 4300 nM T81735 CX8NE4 44421007 IC50 > 30000 nM T81735 CH3L9P 44551660 IC50 = 879 nM T81735 CDZ39K 44562271 IC50 = 370 nM T81735 CYI86D 44562272 IC50 = 480 nM T81735 CBV95H 44562273 IC50 = 240 nM T81735 C0Y1SO 44562274 IC50 = 170 nM T81735 CO9U3W 44562275 IC50 = 1550 nM T81735 C9VFC8 44562319 IC50 = 670 nM T81735 CHQ59J 44562356 IC50 = 300 nM T81735 C0PLB1 44562357 IC50 = 1240 nM T81735 C6WE3Z 44562358 IC50 = 2370 nM T81735 CUW7B0 44562359 IC50 = 1410 nM T81735 CYNE48 44562360 IC50 = 1750 nM T81735 CTGF18 44562385 IC50 = 240 nM T81735 CSP3E8 44562386 IC50 = 510 nM T81735 C03OHZ 44562387 IC50 = 610 nM T81735 CLW0X4 44562388 IC50 = 4450 nM T81735 C80ZTE 44562396 IC50 = 1260 nM T81735 C2Y0IZ 44562453 IC50 = 180 nM T81735 C4U7YZ 44562454 IC50 = 140 nM T81735 C7Y0BH 44562455 IC50 = 830 nM T81735 CZ7E1S 44562456 IC50 = 1480 nM T81735 CWCL48 44562471 IC50 = 1100 nM T81735 CAJ6X4 44562472 IC50 = 1000 nM T81735 C70JNI 44562473 IC50 = 1900 nM T81735 CI4LC8 44562474 IC50 = 510 nM T81735 CD28AS 44562491 IC50 = 260 nM T81735 CJ90XR 44562492 IC50 = 20 nM T81735 C41EQV 44562508 IC50 = 1130 nM T81735 CM4XZ0 44562509 IC50 = 380 nM T81735 C3TD1Y 44562510 IC50 = 270 nM T81735 CNV10L 44562529 IC50 = 1820 nM T81735 C0OQ4B 44562530 IC50 = 1230 nM T81735 CPT5R8 44562531 IC50 = 880 nM T81735 CV05BX 44562551 IC50 = 3050 nM T81735 C8PCS0 44562552 IC50 = 1570 nM T81735 CI9D8W 44562553 IC50 = 400 nM T81735 C1HN4P 44562554 IC50 = 90 nM T81735 CMBQ80 44562588 IC50 = 90 nM T81735 C4W9YI 44562589 IC50 = 2460 nM T81735 CYG3M8 44562590 IC50 = 340 nM T81735 C5HMX7 44562591 IC50 = 710 nM T81735 C90ITS 44608915 IC50 = 2.3 nM T81735 CZH1P9 44609387 IC50 = 3.4 nM T81735 CIMZ27 46198363 IC50 = 1200 nM T81735 CDA3R9 46220225 IC50 = 1020 nM T81735 CU5K1G 46834296 IC50 = 620 nM T81735 CM73PR 46834571 IC50 = 6600 nM T81735 CTO5B6 46834572 IC50 = 740 nM T81735 C5D6RZ 46871847 IC50 = 340 nM T81735 C9WPV7 46871857 IC50 = 330 nM T81735 CQB16A 46872415 Ki > 4000 nM T81735 C6LTZ8 46891211 IC50 = 1800 nM T81735 COI08E 46891212 IC50 = 1200 nM T81735 C6HGY7 46891213 IC50 = 1600 nM T81735 C3M2GW 46891214 IC50 > 10000 nM T81735 C4Z2NA 46891215 IC50 > 10000 nM T81735 C1QGC2 46891259 IC50 > 10000 nM T81735 CVXH10 46891260 IC50 = 1700 nM T81735 CT70HW 46891261 IC50 = 600 nM T81735 COA36T 46891262 IC50 > 10000 nM T81735 CGYB82 46891315 IC50 > 10000 nM T81735 CD3BO4 46891316 IC50 = 2100 nM T81735 CB54XG 46891317 IC50 = 2100 nM T81735 C67SVB 46891318 IC50 = 3200 nM T81735 CLG85W 46891360 IC50 = 2600 nM T81735 CA4J3B 46891361 IC50 = 680 nM T81735 CP2QD0 49784894 IC50 > 10000 nM T81735 C41HJG 49796393 IC50 > 500000 nM T81735 C4VK9F 49843624 IC50 = 1700 nM T81735 CFY13I 49843787 IC50 = 2700 nM T81735 CDO5C6 49843788 IC50 = 1300 nM T81735 CKPA12 49843789 IC50 = 620 nM T81735 CAB0K1 49843943 IC50 = 2500 nM T81735 C5UR4A 49843944 IC50 = 280 nM T81735 CS38FC 49843945 IC50 = 360 nM T81735 CR6XQ7 49843947 IC50 = 4200 nM T81735 CVI0K6 49843948 IC50 = 1200 nM T81735 CUO0D3 49844083 IC50 = 1600 nM T81735 CY8MP7 49867926 IC50 = 150 nM T81735 CKY3V1 50990924 IC50 = 3 nM T81735 CXD71B 51003497 IC50 = 8 nM T81735 CRJ5W8 51358113 IC50 = 0.5 nM T81735 CA50HJ 52915004 Ki = 6 nM T81735 C5R2AH 52937148 IC50 > 8000 nM T81735 CLH8Y5 52937149 IC50 > 8000 nM T81735 CT7X9U 52937150 IC50 > 8000 nM T81735 C12GTQ 52937251 IC50 > 8000 nM T81735 CQ85UH 52937252 IC50 = 5000 nM T81735 CP91TZ 52937253 IC50 = 720 nM T81735 C1MIR4 52937254 IC50 = 2000 nM T81735 CID2E8 52937255 IC50 > 8000 nM T81735 C2H9JY 52937257 IC50 > 8000 nM T81735 CPY82U 52937258 IC50 = 3800 nM T81735 C27QNB 52937357 IC50 = 1400 nM T81735 CFJB79 52937358 IC50 = 2200 nM T81735 CT5K9L 52937359 IC50 = 2200 nM T81735 C85FTW 52937360 IC50 = 4200 nM T81735 CGLT04 52937361 IC50 > 8000 nM T81735 C2ISM3 52937362 IC50 > 8000 nM T81735 C6Q2EN 52937363 IC50 > 8000 nM T81735 CFT9H6 52937453 IC50 > 8000 nM T81735 C4C6DF 52937454 IC50 > 8000 nM T81735 C0T8KI 52937455 IC50 = 1200 nM T81735 CK30PU 52937456 IC50 = 7000 nM T81735 CJU30Y 52937457 IC50 > 8000 nM T81735 C4RJB2 52937458 IC50 > 8000 nM T81735 C69SEB 52937459 IC50 = 2800 nM T81735 CPR6W2 52937553 IC50 > 8000 nM T81735 CQP02L 52937554 IC50 > 8000 nM T81735 CAHU94 52937555 IC50 = 6800 nM T81735 CQ2NU7 52937556 IC50 = 5800 nM T81735 CATX20 52937557 Ki = 2800 nM T81735 CB9WS5 52937558 IC50 > 8000 nM T81735 CUY01F 52937559 IC50 > 8000 nM T81735 CTM68E 52937659 IC50 > 8000 nM T81735 C7G9KF 52937660 IC50 = 3200 nM T81735 C5G6YD 52937661 IC50 = 4400 nM T81735 C6R5OE 52937662 IC50 > 8000 nM T81735 CDHT14 52937663 IC50 = 2100 nM T81735 C0IJZ8 52937664 IC50 = 1400 nM T81735 CGW25Q 52937665 IC50 = 2900 nM T81735 CL04GS 52937759 IC50 = 2400 nM T81735 CU1P2L 52940797 IC50 = 3840 nM T81735 C2KI6V 52942202 IC50 = 10000 nM T81735 CDHJ08 52942235 IC50 = 565 nM T81735 C4VCY0 52943258 IC50 = 1100 nM T81735 C1XEV2 52943394 IC50 = 179 nM T81735 CHI0P6 52944356 IC50 = 860 nM T81735 CU16RS 52944387 IC50 = 1100 nM T81735 CWPC54 52945348 IC50 = 19 nM T81735 C4NLX7 52945630 IC50 = 630 nM T81735 CXD6T8 52945845 IC50 = 1170 nM T81735 C7ET6Z 52948010 IC50 = 85 nM T81735 CV5B2C 52949497 IC50 = 100000 nM T81735 C4J9WZ 53307606 IC50 = 6 nM T81735 C8N5BU 53316474 IC50 = 330 nM T81735 CW8PM0 53317812 IC50 = 12000 nM T81735 C32SJL 53317813 IC50 = 14 nM T81735 CCP80W 53319118 IC50 = 180 nM T81735 C3Z4FD 53320358 IC50 = 1000 nM T81735 CA2QV6 53320444 IC50 = 80 nM T81735 C7C4LR 53320445 IC50 = 3300 nM T81735 C27AWP 53321743 IC50 > 10000 nM T81735 CLX39O 53323075 IC50 = 170 nM T81735 CCP53L 53323076 IC50 = 2600 nM T81735 CP15UQ 53323077 IC50 = 160 nM T81735 CIJ0K1 53323078 IC50 = 110 nM T81735 C7TR8E 53324425 IC50 = 290 nM T81735 C69PLZ 53324426 IC50 = 280 nM T81735 C4CU5V 53325726 IC50 = 500 nM T81735 CUYM86 53326857 IC50 = 690 nM T81735 CW7XT2 53357977 IC50 = 1700 nM T81735 CK43XQ 53358085 IC50 = 330 nM T81735 CEO1V0 53358086 IC50 = 96 nM T81735 C4BJM7 53358087 IC50 = 190 nM T81735 C0Y9ZG 54761473 IC50 > 30000 nM T81735 CT64SR 56599306 IC50 = 4800 nM T81735 CJE64Z 56659562 IC50 = 720 nM T81735 CMY4C6 56663011 IC50 = 930 nM T81735 CF92RJ 56663012 IC50 = 760 nM T81735 C70RYS 56666490 IC50 = 420 nM T81735 CDMI13 56666491 IC50 = 2430 nM T81735 C5GA2X 56669902 IC50 = 3090 nM T81735 C0HNE8 56680036 IC50 = 717 nM T81735 CT6XL0 57466811 IC50 > 10000 nM T81735 C59YAC 57495353 IC50 = 880 nM T81735 C7ONC3 58137106 IC50 = 2700 nM T81735 C8NW9U 59335342 IC50 = 5 nM T81735 CX30US 59335350 IC50 = 6 nM T81735 C1YTI8 59472018 Ki = 8900 nM T81735 C76CVG 59472034 Ki > 4000 nM T81735 C1EW0H 59472203 Ki = 2610 nM T81735 C0MJ3L 59472343 Ki > 4000 nM T81735 CL6F0V 60200387 IC50 = 5 nM T81735 C57DTK 68045182 Ki = 260 nM T81735 CQS8G7 70686830 IC50 > 10000 nM T81735 CS1X6R 71452198 IC50 = 10000 nM T81735 C5P4VC 71452253 IC50 = 5700 nM T81735 CW25OH 71452254 IC50 = 14800 nM T81735 C31VIF 71455748 IC50 = 2500 nM T81735 CA9K1N 71459479 IC50 = 13500 nM T81735 CL26IY 71461215 IC50 = 25200 nM T81735 C3PXR4 71462953 IC50 = 7800 nM T81735 CI1HO0 71521971 Ki > 4000 nM T81735 CI2J9Q 71521995 Ki > 4000 nM T81735 CKB86I 71537083 Ki > 4000 nM T81735 CAVL54 71554734 Ki > 4000 nM T81735 CFR8S3 71817378 IC50 = 24 nM T81735 C2ZIG6 71817379 IC50 = 18 nM T81735 C4OZC1 71817380 IC50 = 8 nM T81735 CWI8P4 71817381 IC50 = 84 nM T81735 CS47OV 71817382 IC50 = 10 nM T81735 CN85GT 71817383 IC50 = 16 nM T81735 CR0PO3 71817384 IC50 = 6 nM T81735 CZ1D3W 71817385 IC50 = 11 nM T81735 C70ZFS 71817542 IC50 = 12 nM T81735 C52JNI 71817543 IC50 = 61 nM T81735 CTRO57 71817544 IC50 = 57 nM T81735 CST61Z 71817699 IC50 = 8 nM T81735 CWX46Q 71817700 IC50 = 43 nM T81735 CGP2L4 71817701 IC50 = 7 nM T81735 CBQ07M 71817854 IC50 = 15 nM T81735 C0F7KZ 71817855 IC50 = 10 nM T81735 C8LSX4 71817856 IC50 = 30 nM T81735 C6T1ON 71818008 IC50 = 13 nM T81735 CMJ3F4 71818009 IC50 = 22 nM T81735 CYS3Z2 71818010 IC50 = 18 nM T81735 CZ74WX 71818011 IC50 = 8 nM T81735 CVIJ19 71818012 IC50 = 9 nM T81735 CZX41G 71818150 IC50 = 37 nM T81735 CPS1L2 71818151 IC50 = 37 nM T81735 C0A4XB 71818152 IC50 = 28 nM T81735 CZ1KP7 71818153 IC50 = 26 nM T81735 C3PI7U 71818154 IC50 = 10 nM T81735 CH8DF3 71818297 IC50 = 22 nM T81735 CWO83Z 71818298 IC50 = 41 nM T81735 CT8A4N 71818299 IC50 = 11 nM T81735 CH03TJ 71818300 IC50 = 9 nM T81735 CGSU20 71818448 IC50 = 12 nM T81735 C21KCX 71818449 IC50 = 6 nM T81735 C3YFK7 71818450 IC50 = 33 nM T81735 C5SEL2 71818451 IC50 = 78 nM T81735 C4CL7G 71818594 IC50 = 31 nM T81735 C0KNP7 71818595 IC50 = 6 nM T81735 C76XIZ 71818596 IC50 = 13 nM T81735 CJX42D 71818724 IC50 = 23 nM T81735 CX4PU2 71818725 IC50 = 19 nM T81735 CLF5Y6 71818726 IC50 = 29 nM T81735 C9YBT3 71818727 IC50 = 33 nM T81735 CCE4L2 71818871 IC50 = 24 nM T81735 CGX4P8 71818872 IC50 = 30 nM T81735 CZOX62 71818873 IC50 = 18 nM T81735 CCJD39 71818874 IC50 = 10 nM T81735 CODJ62 71819011 IC50 = 49 nM T81735 C74VUN 71819012 IC50 = 29 nM T81735 CBZ41O 71819013 IC50 = 42 nM T81735 CTZ0C3 71819014 IC50 = 9 nM T81735 CC36GN 71819149 IC50 = 12 nM T81735 CA21HI 71819150 IC50 = 37 nM T81735 C1SEO5 71819151 IC50 = 8 nM T81735 C8C2BY 71819285 IC50 = 20 nM T81735 C52DAM 71819286 IC50 = 7 nM T81735 C7T4JG 71819287 IC50 = 22 nM T81735 CPT16V 71819288 IC50 = 5 nM T81735 C2WD3L 71819289 IC50 = 10 nM T81735 CZ47NP 71819426 IC50 = 2 nM T81735 CYMO02 71819427 IC50 = 3 nM T81735 CWL72U 71819428 IC50 = 19 nM T81735 C6INP8 71819429 IC50 = 29 nM T81735 CICE45 71819559 IC50 = 44 nM T81735 CS2R7E 71819560 IC50 = 53 nM T81735 CQ4P8O 71819561 IC50 = 61 nM T81735 C2IEY8 71819562 IC50 = 16 nM T81735 CLO1P5 72199292 IC50 > 36 nM T81735 C2HB1D 76313468 IC50 > 10000 nM T81735 C04SRC 77147259 IC50 = 357 nM T81735 CHX2Z3 90435584 Ki = 3350 nM T81735 CF5HV8 118720613 IC50 = 140 nM T81735 C2UIB7 118720614 IC50 = 6500 nM T81735 CSH50J 118720615 IC50 = 1600 nM T81735 C9SF2E 118720891 IC50 > 25000 nM T81735 C81IFQ 122163152 IC50 = 320 nM T81735 C42GSX 122180520 Ki = 1300 nM T81735 CMG21L 122705987 IC50 = 34 nM T81735 CW5EK9 122705988 IC50 = 20300 nM T81735 C2O4RK 127038523 IC50 = 12300 nM T81735 CO27IE 127038894 IC50 = 6050 nM T81735 C72NPR 127039226 IC50 = 7120 nM T81735 CRLD82 127039546 IC50 = 63500 nM T81735 CL0ZU8 127040691 IC50 = 9940 nM T81735 CB0G7Z 127040692 IC50 = 10900 nM T81735 C3ZXT2 127040693 IC50 = 15700 nM T81735 CY6NM3 127040694 IC50 = 8810 nM T81735 C6X0NR 127041034 IC50 = 78400 nM T81735 CLUK47 127042289 IC50 = 269 nM T81735 CZO8N7 127042650 IC50 = 5770 nM T81735 CM9T7X 127042651 IC50 = 564 nM T81735 C05MRE 127042767 IC50 = 9800 nM T81735 C4L9TC 127042949 IC50 = 2120 nM T81735 CVF8Z9 127045862 IC50 = 3 nM T81735 CH68NT 127046076 IC50 = 48 nM T81735 C34REM 127046317 IC50 = 690 nM T81735 CK68CA 130453737 IC50 = 2800 nM T81735 CUO41K 130470684 IC50 = 370 nM T81735 CR4V2T 134140359 IC50 = 1500 nM T81735 CIE64W 134142825 IC50 = 2 nM T81735 CX0UR7 134694318 IC50 = 643 nM T81735 CDQ3V9 135151301 IC50 = 0.1585 nM T81735 C9FUK2 135151360 IC50 = 0.6 nM T81735 CCB30F 135179035 IC50 = 0.3162 nM T81735 CG40SB 135179714 IC50 = 0.07943 nM T81735 CX8AI4 135398491 IC50 = 13 nM T81735 CU29YK 135750268 IC50 = 620 nM T81735 C12UDA 135947972 IC50 = 36 nM T81735 CN42ZS 135947973 IC50 = 190 nM T81735 CF8AO3 135947974 IC50 = 48 nM T81735 CW08GJ 135947976 IC50 = 0.5 nM T81735 C8O9HG 135947977 IC50 = 12000 nM T81735 CJN7E2 135947978 IC50 = 460 nM T81735 CFKH34 135947979 IC50 = 100 nM T81735 C81NTE 135980524 IC50 > 8000 nM T81735 C0AYN4 135980525 IC50 = 1800 nM T81735 CTZA58 137628643 IC50 = 26 nM T81735 CSK0C2 137641008 IC50 = 2 nM T81735 CKDZ26 138504497 IC50 = 1800 nM T81735 C4V1GH 145714280 IC50 = 0.3162 nM T81735 CGA83C 145981271 IC50 > 30000 nM T81735 C5R6BS 145987142 IC50 > 30000 nM T81735 C8X2IT 145996536 IC50 = 1290 nM T81735 CH8J7L 155510809 Ki > 4000 nM T81735 C2MD1Q 155513187 IC50 > 10000 nM T81735 C6ACO5 155513430 IC50 = 2.512 nM T81735 COM30P 155514391 Ki > 4000 nM T81735 CY1B4L 155517765 Ki = 4000 nM T81735 CA6OU5 155520541 IC50 = 10 nM T81735 CIM7F6 155520997 IC50 = 12.59 nM T81735 C2H3ZJ 155521367 IC50 = 0.1995 nM T81735 CH3S0D 155524826 IC50 = 125.89 nM T81735 C23IFK 155526336 IC50 = 1.995 nM T81735 C4NU5J 155532227 IC50 = 10 nM T81735 CSPN68 155532569 Ki = 785 nM T81735 C23IEP 155536557 Ki > 4000 nM T81735 C3TP4A 155537050 IC50 = 3.162 nM T81735 CY32TQ 155537053 IC50 = 0.3981 nM T81735 CP25WZ 155539880 IC50 = 5.012 nM T81735 CBN29V 155544583 IC50 = 109 nM T81735 C9KQT6 155545258 IC50 = 5.012 nM T81735 CHCS54 155546044 Ki > 4000 nM T81735 CQ5OD0 155550395 IC50 = 5 nM T81735 CJ75BO 155552100 IC50 = 204 nM T81735 C2EW5C 155555885 IC50 = 0.2512 nM T81735 CJ9A2Z 155556123 IC50 = 7.943 nM T81735 CO3R8Y 155560892 Ki = 1700 nM T81735 C9KZ5P 155566902 IC50 = 6.31 nM T81735 C1S8ZB 155568922 IC50 = 98 nM T81735 CE6P9C 155569571 Ki > 1600 nM T81735 D00IRL 16745325 IC50 = 220 nM T81735 D00MCG 16203946 IC50 = 400 nM T81735 D00MXW 11609954 IC50 = 14900 nM T81735 D00TUH 11710022 IC50 = 1000 nM T81735 D01MXN 11501108 IC50 = 2600 nM T81735 D01SXB 16203472 IC50 = 2500 nM T81735 D01ZMP 16203941 IC50 = 1100 nM T81735 D02DDM 21106400 IC50 = 380 nM T81735 D02IDN 11471732 IC50 = 7700 nM T81735 D02MPG 10062895 IC50 = 180 nM T81735 D02PBS 11508573 IC50 = 1680 nM T81735 D02SMG 16203943 IC50 = 1000 nM T81735 D02TCZ 11289486 IC50 = 1690 nM T81735 D02TSN 46244454 IC50 > 30000 nM T81735 D03DJC 16203354 IC50 = 7800 nM T81735 D03EHM 24905142 IC50 = 60 nM T81735 D03FTE 16204050 IC50 = 1200 nM T81735 D03IQX 11415057 IC50 = 8590 nM T81735 D03MDA 9965345 IC50 = 650 nM T81735 D03QQH 16760391 IC50 = 270 nM T81735 D04DQF 16203469 IC50 = 4700 nM T81735 D04ECT 11358426 IC50 = 5150 nM T81735 D04JGZ 11709748 IC50 = 1500 nM T81735 D04RAW 11660428 IC50 = 3000 nM T81735 D04SCD 11459783 IC50 = 3270 nM T81735 D04XFN 11566823 IC50 = 4590 nM T81735 D05SBJ 11277489 IC50 = 1900 nM T81735 D05SGV 11437484 IC50 = 1250 nM T81735 D05USL 5278396 IC50 = 183 nM T81735 D06BDY 11196279 IC50 = 1200 nM T81735 D06DAY 11637964 IC50 = 2800 nM T81735 D06GNE 9859309 IC50 = 120 nM T81735 D06TGR 11609490 IC50 = 1200 nM T81735 D06WCT 11624481 IC50 = 2990 nM T81735 D07APP 131255 IC50 = 1260 nM T81735 D07AXO 11346012 IC50 = 10940 nM T81735 D07NSR 11346540 IC50 = 3240 nM T81735 D08BRZ 10912743 IC50 = 350 nM T81735 D08WQW 16203714 IC50 = 800 nM T81735 D09TJK 16203599 IC50 = 3100 nM T81735 D09YAL 16204165 IC50 = 1060 nM T81735 D0AG8B 11174002 IC50 = 1380 nM T81735 D0B0QS 11208656 IC50 = 2010 nM T81735 D0B4CJ 11358716 IC50 = 2240 nM T81735 D0B9EZ 3045697 IC50 = 3810 nM T81735 D0C3SJ 16203712 IC50 = 5900 nM T81735 D0C8MK 11502854 IC50 = 5800 nM T81735 D0D9RN 11715743 IC50 = 450 nM T81735 D0F5BD 25817490 IC50 = 250 nM T81735 D0F6ZC 10083230 IC50 = 1650 nM T81735 D0F7ZK 16203255 IC50 = 4200 nM T81735 D0G0BJ 51000408 IC50 = 26 nM T81735 D0G4RG 11471539 IC50 = 6660 nM T81735 D0H0HR 49836027 IC50 = 6.34 nM T81735 D0H2BL 11522900 IC50 = 380 nM T81735 D0H2CM 135565635 IC50 = 410 nM T81735 D0H9DB 11552705 IC50 = 10600 nM T81735 D0I1LR 11623802 IC50 = 300 nM T81735 D0I7GE 11790 IC50 = 4980 nM T81735 D0J7BH 804048 IC50 = 4820 nM T81735 D0JB6H 11075707 IC50 = 5350 nM T81735 D0K3VK 16203359 IC50 = 2500 nM T81735 D0K5VE 21106425 IC50 = 470 nM T81735 D0K7LZ 11668417 IC50 = 40 nM T81735 D0KG0Z 11471812 IC50 = 5710 nM T81735 D0KH8S 16203474 IC50 = 7200 nM T81735 D0L3TX 686127 IC50 = 8810 nM T81735 D0LC5C 16203826 IC50 = 8100 nM T81735 D0M3RY 21106428 IC50 = 1800 nM T81735 D0N2LW 11324758 IC50 = 1610 nM T81735 D0N2XO 21106405 IC50 = 540 nM T81735 D0O3VF 11602076 IC50 = 700 nM T81735 D0O4KC 11357448 IC50 = 11310 nM T81735 D0O5BC 16204045 IC50 = 800 nM T81735 D0O9OB 11630658 IC50 = 1320 nM T81735 D0P4MU 11529823 IC50 = 8400 nM T81735 D0PO9X 16204046 IC50 = 2300 nM T81735 D0Q4GJ 323484 IC50 = 1920 nM T81735 D0Q5FJ 11185819 IC50 = 4670 nM T81735 D0QB9L 16204047 IC50 = 1300 nM T81735 D0R0TW 11964036 IC50 = 5 nM T81735 D0R1BG 11482391 IC50 = 1200 nM T81735 D0R7HM 10923175 IC50 = 1100 nM T81735 D0S0RK 10680 IC50 > 10000 nM T81735 D0S5SG 16203942 IC50 = 1600 nM T81735 D0S5YV 6852167 IC50 = 64 nM T81735 D0S7NM 11652716 IC50 = 2600 nM T81735 D0T0BY 10039361 IC50 = 280 nM T81735 D0T9DI 3163532 IC50 > 10000 nM T81735 D0U7WU 11437483 IC50 = 390 nM T81735 D0U9ZW 10857738 IC50 = 8050 nM T81735 D0V0SD 269395 IC50 = 2000 nM T81735 D0V3XZ 11515664 IC50 = 2400 nM T81735 D0V8VY 3045696 IC50 = 6170 nM T81735 D0W1ST 9860529 IC50 = 230 nM T81735 D0W3QB 11426483 IC50 = 260 nM T81735 D0W8XH 9884685 IC50 = 14 nM T81735 D0X7TB 10017389 IC50 = 190 nM T81735 D0Y3OO 11327430 Ki = 0.65 nM T81735 D0Y7WU 21106426 IC50 = 530 nM T81735 D0Z2CN 135418335 IC50 = 10000 nM T81735 D0Z3CC 16204049 IC50 = 900 nM T81735 D0ZQ8Z 11448366 IC50 = 950 nM T00602 D00ENY 33032 IC50 = 11000 nM T00602 C9CQV1 131738 IC50 = 270000 nM T00602 C7BKY8 164701 IC50 = 100000 nM T00602 C45TML 1755783 IC50 > 300000 nM T00602 CDK9W5 1796705 IC50 > 300000 nM T00602 C8L6JU 2177697 IC50 = 22908.68 nM T00602 CRQW20 2266743 IC50 > 300000 nM T00602 CO0I2U 2266913 IC50 > 300000 nM T00602 C9HE6N 2271641 IC50 > 300000 nM T00602 CH4RP6 2271698 IC50 > 300000 nM T00602 C3SL4Y 2271738 IC50 > 300000 nM T00602 C7K9MX 2283576 IC50 = 12000 nM T00602 CB6EZ4 2285406 IC50 > 300000 nM T00602 CBW36C 2287441 IC50 > 316227.77 nM T00602 C13DLB 2289587 IC50 > 316227.77 nM T00602 CZQ83G 2289624 IC50 > 300000 nM T00602 CFG35Z 2737891 IC50 = 2290.87 nM T00602 CYR4X2 2838960 IC50 = 3630.78 nM T00602 CP4L3M 2839392 IC50 = 4000 nM T00602 CF2LE3 4133412 IC50 = 3162.28 nM T00602 CJW9P4 5506801 IC50 > 300000 nM T00602 C5PWJ3 6505351 IC50 > 300000 nM T00602 CTBZ42 6505352 IC50 = 100000 nM T00602 C64QSY 7016554 Ki = 11481.54 nM T00602 CTMP80 9920506 Ki = 22908.68 nM T00602 C2EA8S 10219727 IC50 > 1000000 nM T00602 C53YBE 10419887 Ki > 400000 nM T00602 C2PE4O 10464763 IC50 = 100000 nM T00602 C46KUE 10680281 Ki = 117489.76 nM T00602 C2WQB7 10877814 IC50 > 1000000 nM T00602 C83OPZ 10954230 IC50 > 1000000 nM T00602 C7Z6AX 10986716 IC50 > 1000000 nM T00602 C78YAI 10997729 IC50 > 1000000 nM T00602 CE80SU 11041159 IC50 > 1000000 nM T00602 CMSD95 11062853 IC50 > 1000000 nM T00602 C2TWR9 11063103 IC50 > 1000000 nM T00602 C0HT8M 11528550 Ki = 40738.03 nM T00602 CQ5H1B 11543205 Ki = 127000 nM T00602 C2QJU5 11616374 IC50 = 2000 nM T00602 CZ9V5S 11629898 Ki = 28840.32 nM T00602 C5E8BT 11651356 Ki = 47863.01 nM T00602 CV76LO 11667702 IC50 = 3800 nM T00602 C7SHB1 11745400 Ki = 10232.93 nM T00602 C0BM2Z 12047098 IC50 = 69000 nM T00602 C68AOJ 12047099 IC50 = 15000 nM T00602 C09XIT 12047100 IC50 = 16000 nM T00602 C1X3YB 16727662 IC50 > 300000 nM T00602 C6XLF5 24905646 IC50 = 3000000 nM T00602 CFI54P 24905647 IC50 > 1000000 nM T00602 CQK96U 24905648 IC50 > 3000000 nM T00602 C36NMZ 24905649 IC50 = 1000000 nM T00602 CB3T7C 24905650 IC50 = 1000000 nM T00602 C14RNW 24905651 IC50 = 3000000 nM T00602 CM1S2B 24905652 Ki = 450000 nM T00602 CUS45D 24905703 IC50 > 3000000 nM T00602 C86BUK 24905705 Ki > 3000000 nM T00602 CJ25EZ 44404580 IC50 = 300 nM T00602 C0LJ8T 44404590 IC50 = 3000 nM T00602 CJD1V7 44404611 IC50 = 700 nM T00602 CJ6ER9 44404615 IC50 = 2000 nM T00602 C4CZN1 44405320 Ki = 28840.32 nM T00602 C8TMX2 44417425 Ki = 200000 nM T00602 CYQ2S5 49782834 IC50 > 1000000 nM T00602 C94ZJF 49782835 IC50 > 100000 nM T00602 CZ5YU8 49783035 IC50 > 100000 nM T00602 CR2IM7 49910175 IC50 > 316227.77 nM T00602 CY91US 52941382 IC50 = 3.548 nM T00602 CI76TC 70688590 IC50 > 300000 nM T00602 C2J4MG 70690647 IC50 > 300000 nM T00602 C4HI0U 70789291 IC50 > 3000000 nM T00602 CP48NY 71449125 IC50 = 20000 nM T00602 C7NYC0 71449126 IC50 = 2000 nM T00602 CD03AH 71449127 IC50 = 700 nM T00602 CVST26 71450915 IC50 = 150 nM T00602 C31HCW 71450916 IC50 = 1000 nM T00602 CC15SM 71450917 IC50 = 100000 nM T00602 CBZ9D6 71450918 IC50 = 22000 nM T00602 CSO9P3 71452727 IC50 = 200 nM T00602 C23DMA 71452728 IC50 = 130 nM T00602 CE0A3V 71452729 IC50 = 6000 nM T00602 CRKN62 71452730 IC50 = 2900 nM T00602 C8X4VU 71454504 IC50 = 200 nM T00602 COUY80 71454505 IC50 = 100 nM T00602 C8QW6K 71454506 IC50 = 1000 nM T00602 CKWF24 71454507 IC50 = 6000 nM T00602 CDY5K2 71456248 IC50 = 400 nM T00602 C9O7LC 71456249 IC50 = 100 nM T00602 C1HJF2 71458054 IC50 = 300 nM T00602 C3P0MQ 71461655 IC50 = 3000 nM T00602 C0P4NT 71574743 IC50 > 300000 nM T00602 CGH79X 71574744 IC50 > 300000 nM T00602 COC8W2 71574746 IC50 > 300000 nM T00602 C5U9HZ 71574747 IC50 > 300000 nM T00602 C35BOJ 71574834 IC50 > 1000000 nM T00602 CNVG02 71574836 IC50 = 100000 nM T00602 C2JS0I 71574837 IC50 = 200000 nM T00602 CV5IT8 71574838 IC50 > 1000000 nM T00602 CL9BJ8 71574839 IC50 > 1000000 nM T00602 CCS4T2 71574840 IC50 > 1000000 nM T00602 CM5Z0I 71574841 IC50 > 300000 nM T00602 C3Z0TH 73348758 Ki = 200000 nM T00602 C8DGU5 90480101 IC50 > 1000000 nM T00602 CEH82V 90480134 IC50 > 1000000 nM T00602 CT2KF1 127030385 IC50 > 300000 nM T00602 CX95LC 127030386 IC50 > 300000 nM T00602 C8TS1X 127030387 IC50 > 300000 nM T00602 CF6NI8 127031290 IC50 > 300000 nM T00602 C2V5PM 132820245 IC50 = 31 nM T00602 CC54HS 134131748 IC50 = 31622.78 nM T00602 CM8O9I 134131963 IC50 = 794.33 nM T00602 C26CTG 134132565 IC50 = 199526.23 nM T00602 CGXV98 134133631 IC50 = 9332.54 nM T00602 C1ZAB4 134134123 IC50 = 70000 nM T00602 CZ2WH5 134134813 IC50 = 4000 nM T00602 CT3MU6 134135313 IC50 = 300000 nM T00602 CTL6A4 134135682 IC50 = 49000 nM T00602 C0MJT1 134136786 IC50 = 100000 nM T00602 CA40DU 134137403 IC50 = 12882.5 nM T00602 C1L9UX 134139672 IC50 = 1700 nM T00602 CC24GI 134139698 IC50 > 1000000 nM T00602 CTSA19 134139982 IC50 = 2500 nM T00602 CWS62H 134140412 IC50 = 43651.58 nM T00602 C5QIB1 134140490 IC50 = 63000 nM T00602 CT4QN8 134141720 IC50 = 8800 nM T00602 CJF5X7 134143016 IC50 = 300000 nM T00602 C4CT5L 134144465 IC50 = 1949.84 nM T00602 CL0EA9 134144947 IC50 = 16000 nM T00602 COM76W 134147363 IC50 > 300000 nM T00602 C9Q2JY 134147568 IC50 = 2300 nM T00602 CS38BI 134147884 IC50 = 3800 nM T00602 CP10YS 134148109 IC50 = 100000 nM T00602 CTPS85 134149212 IC50 = 2700 nM T00602 COP15G 134149427 IC50 = 2238.72 nM T00602 C6HQS8 134149488 IC50 = 794.33 nM T00602 CTH41F 134149576 IC50 = 18000 nM T00602 CQ8R9N 134149841 IC50 = 64565.42 nM T00602 C10RSO 134150446 IC50 > 300000 nM T00602 C9N0CQ 134152035 IC50 = 300000 nM T00602 C5SN8C 134152143 IC50 = 350 nM T00602 C3RAO8 134153858 IC50 = 380 nM T00602 CI3HS7 134155673 IC50 = 316.23 nM T00602 CVT7Q4 134157558 IC50 = 1600 nM T00602 CHK48B 137643975 IC50 > 1000000 nM T00602 C6J8RH 137658224 IC50 > 1000000 nM T00602 CS1X0H 145952067 IC50 = 6.1 nM T00602 C2X6ST 145952092 IC50 = 1659.59 nM T00602 CRXG02 145952717 IC50 = 2691.53 nM T00602 CZD62V 145953140 IC50 = 3000 nM T00602 C5SH4V 145953224 IC50 = 99000 nM T00602 C63MDC 145954707 IC50 = 20.89 nM T00602 C87HDC 145955435 IC50 = 6900 nM T00602 CT3H6G 145955563 IC50 = 1600 nM T00602 CIN7D3 145955863 IC50 = 1380.38 nM T00602 CZ7N3B 145956590 IC50 = 620 nM T00602 CFZK42 145957754 IC50 = 1200 nM T00602 CEX81Q 145958688 IC50 = 87000 nM T00602 C6BP3Z 145959256 IC50 = 2200 nM T00602 C8DIJ6 145960111 IC50 = 3400 nM T00602 CET93L 145971223 IC50 = 1.259 nM T00602 CGF5S1 145971489 IC50 = 29000 nM T00602 C30JVP 145971753 IC50 = 1258.93 nM T00602 CI04HT 145972021 IC50 = 11.75 nM T00602 C18GNB 145973375 IC50 = 10.72 nM T00602 CK7UW9 155519942 IC50 > 300000 nM T00602 C0Y9UF 155520160 IC50 > 300000 nM T00602 C52DFC 155524441 IC50 = 10715.19 nM T00602 C4IWE9 155525454 IC50 > 316227.77 nM T00602 CHJ5G1 155527881 IC50 > 316227.77 nM T00602 C9Z2ME 155529757 IC50 = 38000 nM T00602 CN1S4G 155530850 IC50 > 316227.77 nM T00602 C7HOI6 155533200 IC50 > 300000 nM T00602 CG65QS 155536541 IC50 = 34673.69 nM T00602 CX3ED4 155538143 IC50 > 300000 nM T00602 C4J3DC 155541203 IC50 = 100000 nM T00602 CD4B0V 155542542 IC50 > 300000 nM T00602 C87POT 155548017 IC50 > 300000 nM T00602 CPQM13 155555116 IC50 > 300000 nM T00602 CV9R4S 155557780 IC50 > 316227.77 nM T00602 C6NAQ5 155561202 IC50 > 300000 nM T00602 CF9YI6 155564787 IC50 > 300000 nM T00602 CFN45I 155565203 IC50 > 300000 nM T00602 CCK6T7 155565355 IC50 = 15848.93 nM T00602 D02JJX 11531745 IC50 = 5000 nM T00602 D03RGP 1221 IC50 > 1000000 nM T00602 D03UIR 24905704 IC50 = 1000000 nM T00602 D04XZP 107883 IC50 > 3000000 nM T00602 D07GUB 5311218 IC50 = 1621.81 nM T00602 D09HET 11622683 IC50 = 51000 nM T00602 D0F5SO 11369932 IC50 = 300 nM T00602 D0JT2N 443239 IC50 = 3890.45 nM T00602 D0OT9B 5960 IC50 = 9300 nM T00602 D0X3CF 442879 IC50 > 500000 nM T76414 D0I0DL 3689 Ki = 10 nM T76414 D04WUA 219101 IC50 = 74 nM T76414 D0S8CI 60703 Ki = 13 nM T76414 D06RCS 156328 Ki = 30 nM T76414 D0K0DB 6604887 IC50 = 9 nM T76414 D0LD9S 1103 EC50 = 125000 nM T76414 C63KYD 66637 IC50 = 9400 nM T76414 CTO7F3 200369 Ki = 10000 nM T76414 C57RKT 610414 IC50 > 10000 nM T76414 CMNK42 659834 IC50 > 10000 nM T76414 CD48TY 694463 IC50 = 90000 nM T76414 CH73AF 913218 IC50 = 769 nM T76414 C5G4FA 1394668 IC50 = 7.943 nM T76414 C8QPT9 2806914 IC50 = 720 nM T76414 C5Z6NT 3113150 IC50 = 78000 nM T76414 CXF09D 4231127 EC50 > 10000 nM T76414 CN85UI 4235339 IC50 = 113000 nM T76414 CIA9B5 9794218 IC50 > 300000 nM T76414 C4VS0G 9797323 IC50 = 4.1 nM T76414 CUGX54 9797385 EC50 = 1.6 nM T76414 C8V2ZD 9799094 Ki = 12 nM T76414 CL79YZ 9858476 Ki = 180 nM T76414 C8XZ9O 9862028 IC50 = 9.7 nM T76414 CD98TS 9862575 Ki = 3.6 nM T76414 CJ7Q4Y 9863769 IC50 = 47 nM T76414 CKI48D 9878031 Ki = 9 nM T76414 C7D9GT 9881090 Ki = 3.4 nM T76414 C67VXG 9904185 IC50 = 46 nM T76414 C29WVT 9923385 Ki = 23 nM T76414 CAPM04 9927159 Ki = 1.2 nM T76414 C18CEH 9927645 Ki = 2 nM T76414 CC9IL5 9928952 Ki = 0.6 nM T76414 CEB1I2 9945500 Ki = 190 nM T76414 CKLH03 9967123 Ki = 14 nM T76414 C10ROQ 9972103 IC50 = 70 nM T76414 C09KVR 9972180 IC50 = 130 nM T76414 C3TL5R 10018269 IC50 = 9 nM T76414 CD75GU 10131619 Ki = 122 nM T76414 C4KU1Y 10268204 Ki = 37 nM T76414 CU1ZW4 10268255 Ki = 75 nM T76414 C8K2SI 10269028 Ki = 18 nM T76414 C95QAN 10313748 IC50 = 27 nM T76414 CGUQ10 10425979 IC50 = 35 nM T76414 C4MCK2 10426105 IC50 = 100 nM T76414 CQ9NP6 11198145 Ki = 10 nM T76414 CZ8E3X 11771731 Ki = 10 nM T76414 C3CID8 12045491 IC50 = 4300 nM T76414 C4Z0SE 12045492 IC50 = 630 nM T76414 CN6RL1 12045493 IC50 = 610 nM T76414 CJ0EZ4 12045494 IC50 = 1000 nM T76414 CM1S6P 12045495 IC50 = 560 nM T76414 C13FGE 12045496 IC50 = 6400 nM T76414 CYL2J7 12045497 IC50 = 910 nM T76414 CRB59C 12045498 IC50 = 1000 nM T76414 C27OQJ 12045832 IC50 = 930 nM T76414 CO31ZL 15061905 Ki = 16 nM T76414 C1AMD7 16109385 Ki = 220 nM T76414 CKH4Z6 16109388 Ki = 227 nM T76414 CF0RV8 16109389 Ki = 540 nM T76414 CN4BI3 16109390 Ki = 23 nM T76414 CG4BW9 16109391 Ki = 18 nM T76414 CW39HA 16109392 Ki = 150 nM T76414 C3FOV2 16109394 Ki = 227 nM T76414 CES20L 16109395 Ki = 7.8 nM T76414 CR5XJ1 16109396 Ki = 460 nM T76414 CL3OT7 16109399 Ki = 310 nM T76414 CGYP24 16109400 Ki = 1170 nM T76414 CGQ61S 16109401 Ki = 266 nM T76414 C9V1FE 16109406 Ki > 15000 nM T76414 CM54QA 16109414 Ki = 2100 nM T76414 CAC6U1 16109416 Ki = 7400 nM T76414 CZ7P5I 16109418 Ki = 206 nM T76414 C1PM2V 16109419 Ki = 3.7 nM T76414 CBS3C5 16109420 Ki = 720 nM T76414 CH0RU2 20706422 Ki = 16 nM T76414 CT96JI 20706430 IC50 = 420 nM T76414 CM84AP 20706433 Ki = 63 nM T76414 CB0Q1R 20706457 Ki = 2000 nM T76414 CZFK48 20706461 IC50 = 450 nM T76414 C1HV2R 20706464 Ki = 4200 nM T76414 C6NW9F 20706471 Ki = 1800 nM T76414 CGFD68 22240172 IC50 = 12 nM T76414 CDUS81 22273748 Ki = 6.9 nM T76414 CI28HT 22432385 EC50 = 15700 nM T76414 C4RV3J 22499189 Ki = 57 nM T76414 C3BC8U 22616316 Ki = 8 nM T76414 CY0BC7 34924882 IC50 = 210 nM T76414 CA72VD 44322229 IC50 = 38000 nM T76414 CQ21VN 44365962 IC50 = 100 nM T76414 CDZ04W 44366039 IC50 = 380 nM T76414 CCJD07 44366045 IC50 = 240 nM T76414 C4BJ6F 44366056 IC50 = 7400 nM T76414 CR84AS 44366090 IC50 = 1600 nM T76414 C4DL5Q 44366109 IC50 = 150 nM T76414 CRA24L 44366153 IC50 = 630 nM T76414 C9CX5W 44366275 IC50 = 4800 nM T76414 C43JWL 44374616 Ki = 3.9 nM T76414 C5K1IT 44374617 IC50 = 660 nM T76414 CCNK41 44374627 Ki = 20 nM T76414 C9UAG5 44374660 IC50 = 48 nM T76414 CEO8L5 44374667 Ki = 1100 nM T76414 C3X8AB 44374891 Ki = 3500 nM T76414 C0BA2Q 44374892 IC50 = 360 nM T76414 CKB0W3 44374973 Ki = 3900 nM T76414 CDI2T8 44375002 Ki > 15000 nM T76414 CV4X2U 44419241 Ki = 1250 nM T76414 C27AGQ 44419261 Ki = 3100 nM T76414 CQAD48 44419263 Ki = 3180 nM T76414 CA2ST1 44441266 Ki = 7350 nM T76414 CRDB57 44441267 Ki = 4197 nM T76414 CVQG48 44441268 Ki = 296 nM T76414 CXMC83 44441269 Ki = 66 nM T76414 CEMD86 44441270 Ki = 223 nM T76414 CBLS43 44441271 Ki = 75 nM T76414 CYL47C 44441272 Ki = 353 nM T76414 C7Y1LT 44441273 Ki = 505 nM T76414 CF6HC7 44441274 Ki = 2.2 nM T76414 C3UXI0 46845430 Ki = 5.4 nM T76414 CIC1G6 46861929 IC50 = 193000 nM T76414 CG3LA9 53248849 IC50 = 770 nM T76414 CQ0YA3 54581861 IC50 = 508 nM T76414 CB8JV7 54582823 IC50 = 262 nM T76414 C8MH6B 54587759 IC50 = 673 nM T76414 C4KWB0 56654447 EC50 = 34000 nM T76414 C7XPS1 66727815 IC50 = 2400 nM T76414 C0OEX6 70680972 IC50 = 79.43 nM T76414 C3HVG7 70680973 IC50 = 2511.89 nM T76414 CV0D9J 70681106 IC50 = 251.19 nM T76414 C7H4LI 70681107 IC50 = 630.96 nM T76414 C9HQ7U 70683093 IC50 > 10000 nM T76414 CQRZ75 70683233 IC50 = 39.81 nM T76414 CHFM92 70685176 IC50 = 398.11 nM T76414 CG6BY1 70685177 IC50 = 79.43 nM T76414 C3R2JX 70685326 IC50 = 7.943 nM T76414 CSZW57 70687333 IC50 = 1584.89 nM T76414 CE4B9K 70687334 IC50 = 1000 nM T76414 CLJ36Y 70687463 IC50 = 794.33 nM T76414 COXD69 70689390 IC50 = 794.33 nM T76414 CKLR07 70691639 IC50 = 7.943 nM T76414 CQ0IJ9 70691640 IC50 = 39.81 nM T76414 CB6FW9 70691641 IC50 = 398.11 nM T76414 CF2MP0 70693725 IC50 = 31.62 nM T76414 C1FL8O 70695707 IC50 = 199.53 nM T76414 C47ZED 70695843 IC50 = 79.43 nM T76414 CI3X6S 70695844 IC50 = 12.59 nM T76414 CA3H2I 70695845 IC50 = 39.81 nM T76414 CT54NB 86302361 Ki = 10 nM T76414 CC9B6T 91820646 Ki = 6.3 nM T76414 C85CMJ 101884136 Ki = 20 nM T76414 CA83QV 101884137 Ki = 17 nM T76414 CCL4Q7 101884138 Ki = 2.3 nM T76414 CK9JC5 101884139 Ki = 12 nM T76414 CRK6M1 101884140 Ki = 2.9 nM T76414 CG84LB 118207404 IC50 = 4.2 nM T76414 CZ4MS7 118722423 Ki = 16 nM T76414 CFM30P 118864208 IC50 = 3700 nM T76414 C6L4OC 118864285 IC50 = 2460 nM T76414 C9DM5W 118864313 IC50 = 890 nM T76414 CF09GY 118864337 IC50 = 370 nM T76414 C8AR7P 118864437 IC50 = 230 nM T76414 CS20BC 118864476 IC50 = 1750 nM T76414 C4D9VF 118864482 IC50 = 350 nM T76414 C3J1MU 127034644 Ki = 7.6 nM T76414 CN1S8B 127034645 Ki = 3.3 nM T76414 C50RHS 127034646 Ki = 1.6 nM T76414 C4HC6A 127037642 Ki = 3.8 nM T76414 CN03DF 127045755 Ki = 697 nM T76414 C6E8BS 145949157 Ki = 31 nM T76414 CAB3N0 145950456 Ki = 65 nM T76414 CJ89WR 145954168 Ki = 34 nM T76414 C9X4EA 145957598 Ki = 54 nM T76414 CAQ85J 145990650 Ki = 28 nM T76414 CO5UX1 145990703 Ki = 186 nM T76414 C4S9HQ 145991009 Ki = 21 nM T76414 C68VDU 145991437 Ki = 17 nM T76414 CN50PL 145991874 Ki = 27 nM T76414 C1DB5H 145992688 IC50 = 12 nM T76414 C8IWU3 145993787 Ki = 101 nM T76414 CB4H9Y 145993832 Ki = 16 nM T76414 CHC6M2 155513921 Ki = 193 nM T76414 C61VMR 155535499 Ki = 460 nM T76414 CME7I4 155539094 Ki = 204 nM T76414 C5PC6O 155563006 Ki = 128 nM T76414 CW9H1B 155564060 Ki = 26 nM T76414 C1QOX5 155567776 Ki = 48 nM T76414 D06XGK 105074 EC50 = 33000 nM T76414 D07SGS 44292136 Ki = 93 nM T76414 D09HXX 4787937 IC50 > 10000 nM T76414 D0IO8J 3025961 IC50 = 18000 nM T76414 D0K7EZ 9900027 Ki = 0.7 nM T83382 CJY35N 10102480 EC50 = 0.5754 nM T83382 CTE84B 10260704 IC50 = 0.29 nM T83382 CRF1I2 10351235 EC50 = 0.45 nM T83382 CK56IA 13920660 EC50 = 18.6 nM T83382 C39FCZ 13920665 EC50 = 3171 nM T83382 CZM45J 13920666 EC50 = 683.7 nM T83382 CH82QU 13920670 IC50 = 775.5 nM T83382 CO7X1P 45277088 Ki < 10000 nM T83382 C26EWX 45277089 Ki < 10000 nM T83382 C6X4ER 45277090 Ki < 10000 nM T83382 CH7I1J 45277245 Ki < 10000 nM T83382 C8FO0Q 87415277 EC50 = 9.5 nM T83382 C4LZ8G 87415284 EC50 = 7.8 nM T83382 CMFU53 88563444 EC50 = 2.7 nM T83382 C4QSN7 102340758 IC50 = 4286 nM T83382 COA2W3 117072558 EC50 = 0.083 nM T83382 CAX3W4 118708073 EC50 = 9 nM T83382 CGH1K9 118708139 EC50 = 0.14 nM T83382 CT7E1P 118721282 EC50 = 709.4 nM T83382 CFH73K 126558991 EC50 = 12.3 nM T83382 C4LTY5 127025171 EC50 = 162.18 nM T83382 C2Y8WJ 127025772 EC50 = 1348.96 nM T83382 C4B7GF 127026380 EC50 = 141.25 nM T83382 CS7H6Y 127026692 EC50 = 5011.87 nM T83382 C39QJN 127026693 EC50 = 58.88 nM T83382 CS4M3H 127027325 EC50 = 12589.25 nM T83382 CDA87B 127028302 EC50 = 0.5623 nM T83382 C09HYQ 127029245 EC50 = 47.86 nM T83382 C7PDT0 137633449 EC50 = 0.32 nM T83382 CAYE32 137633990 EC50 > 1000 nM T83382 C3UFT4 137634009 EC50 = 0.17 nM T83382 C9J6MS 137634038 EC50 > 1000 nM T83382 C4MP6D 137635007 EC50 = 2.2 nM T83382 CV0SA3 137635179 EC50 > 1000 nM T83382 C9A1NV 137636126 EC50 = 39 nM T83382 CZ4ER6 137636135 EC50 > 1000 nM T83382 CEZI98 137636174 EC50 > 1000 nM T83382 C0V4QH 137636908 EC50 = 1.3 nM T83382 CI3EN9 137637194 EC50 = 0.73 nM T83382 CO5KI9 137638792 EC50 > 1000 nM T83382 CI8Z6A 137639361 EC50 = 100 nM T83382 C60GTH 137639547 EC50 = 49 nM T83382 CZA43W 137640394 EC50 = 81 nM T83382 CH0M4E 137640682 EC50 = 0.77 nM T83382 C8EPD9 137640690 EC50 = 9.5 nM T83382 C3SY4E 137640722 EC50 = 45 nM T83382 C0BR5G 137642468 EC50 > 1000 nM T83382 C1NZS2 137642598 EC50 > 1000 nM T83382 CEZO84 137642989 EC50 = 0.41 nM T83382 C8Z5TV 137643044 EC50 = 2.7 nM T83382 C6D5PN 137643754 EC50 = 17 nM T83382 C62VJS 137643907 EC50 = 1.9 nM T83382 CZW4O1 137644441 EC50 = 34 nM T83382 C7LTU5 137645284 EC50 = 6.3 nM T83382 CB4PL6 137646480 EC50 > 1000 nM T83382 CA91FH 137646678 EC50 = 9.2 nM T83382 CY9VN0 137647003 EC50 > 1000 nM T83382 C9SRK0 137647843 EC50 = 25 nM T83382 CMZO51 137651400 EC50 = 67 nM T83382 C6BZ4Q 137652197 EC50 = 34 nM T83382 C4IZF9 137652435 EC50 = 1 nM T83382 C41GTA 137652696 EC50 = 0.96 nM T83382 C02CQP 137652739 EC50 = 200 nM T83382 CX1O2U 137654882 EC50 = 31 nM T83382 C2GCF6 137654963 EC50 = 48 nM T83382 C23CJO 137656685 EC50 = 52 nM T83382 CS7M0W 137657007 EC50 = 0.25 nM T83382 CIOB49 137657622 EC50 = 42 nM T83382 CHVG89 137660286 EC50 = 42 nM T83382 C1PA4N 137660608 EC50 = 32 nM T83382 CC0DM7 137660871 EC50 = 0.31 nM T83382 C3U2AG 137662007 EC50 = 8.1 nM T83382 CXU43I 145948899 EC50 = 1.778 nM T83382 CGC6I4 145948939 EC50 = 7943.28 nM T83382 CJ90ZA 145948940 EC50 = 128.82 nM T83382 C1XUP6 145948945 EC50 = 6309.57 nM T83382 CXL19B 145948995 EC50 = 1348.96 nM T83382 C6T9KU 145949005 EC50 = 501.19 nM T83382 CI3CP8 145949312 IC50 = 162.3 nM T83382 CJE9N8 145949890 IC50 = 0.34 nM T83382 CMXF70 145950449 EC50 = 8.1 nM T83382 C08LUS 145950548 EC50 = 184.9 nM T83382 C7HT6J 145950907 IC50 = 350.1 nM T83382 CJX82E 145950926 IC50 = 83.1 nM T83382 CH40RP 145951399 EC50 = 343.4 nM T83382 CH9E5Y 145951684 EC50 = 5.1 nM T83382 CE0H7Z 145952282 IC50 = 2.4 nM T83382 C5JNT2 145952841 IC50 = 62.9 nM T83382 C13JWO 145953216 EC50 = 191.7 nM T83382 CN17CJ 145953723 EC50 = 28.8 nM T83382 C1VAK6 145953783 EC50 = 230 nM T83382 CYXG32 145954208 IC50 = 0.54 nM T83382 C0PZ9I 145954222 EC50 = 5.5 nM T83382 CJ9IZ8 145954330 IC50 = 1.6 nM T83382 C5WO9C 145955290 IC50 = 1.2 nM T83382 CSZR24 145955540 IC50 = 8.6 nM T83382 CMVI71 145956001 EC50 = 1053 nM T83382 CJ1FS2 145956177 IC50 = 8.2 nM T83382 C5C9QN 145956751 IC50 = 0.88 nM T83382 C4EKH3 145957679 IC50 = 173.8 nM T83382 C3LE8D 145958000 IC50 = 0.092 nM T83382 C80IPJ 145958151 IC50 = 0.31 nM T83382 C0YGX7 145958189 IC50 = 28.1 nM T83382 CN9M8W 145958420 IC50 = 844.4 nM T83382 C7R5OF 145958560 IC50 = 3755 nM T83382 CS3DU2 145958712 EC50 = 28.5 nM T83382 CQ23YK 145959083 IC50 = 100.1 nM T83382 C8KW6U 145959164 EC50 = 93 nM T83382 C3P6KU 145959336 IC50 = 3 nM T83382 CPS2V1 145959590 IC50 = 37 nM T83382 CM8EN5 145959730 EC50 = 216.6 nM T83382 CC6I9T 145959831 IC50 = 0.36 nM T83382 C0XDK3 145959870 EC50 = 10.9 nM T83382 COJ4G1 145960270 EC50 = 65.8 nM T83382 CZYI89 145960563 IC50 = 0.41 nM T83382 C48HCB 145971434 EC50 = 4.2 nM T83382 C3F4IC 145971940 IC50 = 18320 nM T83382 CEFK04 145972185 IC50 = 0.51 nM T83382 CX6Q5M 145972641 EC50 = 843 nM T83382 CXS39Z 145972936 IC50 = 0.15 nM T83382 CQ3M5K 145973626 EC50 = 273.2 nM T83382 C9IJP3 145974070 EC50 = 822.7 nM T83382 C12QJH 145974338 EC50 = 274.6 nM T83382 D0M9DD 91623352 EC50 = 2.2 nM T50773 D02EYG 10096344 IC50 > 100000 nM T50773 D0K9MY 11243969 IC50 > 30000 nM T50773 D0L3DK 6918537 IC50 > 20000 nM T50773 D0NJ5H 11450633 IC50 > 100000 nM T50773 D0T8XB 44513473 IC50 = 176700 nM T50773 D0U2JP 4369359 IC50 = 59830 nM T50773 D04XIO 11253490 IC50 > 400 nM T50773 D07HZG 11516136 IC50 = 3300 nM T50773 D0FQ2U 6918572 IC50 = 15 nM T50773 D0M3XR 46209133 IC50 > 67000 nM T50773 D0R9HL 11077541 IC50 = 210000 nM T50773 D05FMP 66561557 IC50 > 100000 nM T50773 D07JHU 71667377 IC50 > 100000 nM T50773 D0C6NX 73356493 IC50 > 100000 nM T50773 D0QX2U 71667229 IC50 > 100000 nM T50773 D00FYF 9796290 IC50 = 26250 nM T50773 D0A1NU 16049769 Ki > 30000 nM T50773 CT2EY7 56877 IC50 > 100000 nM T50773 CPEY84 688304 IC50 > 100000 nM T50773 CT2CQ8 3021908 IC50 = 79000 nM T50773 CX08LH 3081017 IC50 > 100000 nM T50773 CAZ25S 3318661 IC50 = 55300 nM T50773 C4RE5F 7020797 IC50 = 79000 nM T50773 C14VRG 9794073 IC50 = 145000 nM T50773 CQT36A 9794235 IC50 = 28000 nM T50773 CSA6V9 9796352 Ki = 24700 nM T50773 CUNB40 9817010 IC50 = 2.03 nM T50773 CKR9Y5 9823963 IC50 = 1600 nM T50773 C8EK7G 9835053 IC50 > 100000 nM T50773 CW5EZ7 9835382 IC50 > 100000 nM T50773 CV87XC 9835734 Ki > 22385 nM T50773 CAHB35 9836210 IC50 = 50000 nM T50773 CUD46C 9855673 IC50 = 152000 nM T50773 C8XO1Z 9859008 Ki > 22385 nM T50773 C5CZ6J 9865563 Ki > 22385 nM T50773 CR9AW7 9870934 IC50 = 280 nM T50773 C2TV9M 9884543 IC50 = 2.7 nM T50773 CMGX12 9920733 IC50 = 1160 nM T50773 C4EC8A 9924995 IC50 = 23000 nM T50773 CFH1V2 9942336 IC50 = 130 nM T50773 C28XTC 9942425 IC50 > 1000000 nM T50773 CZ1S9O 9942554 IC50 = 21 nM T50773 CZMT26 9947730 IC50 > 100000 nM T50773 CLR78W 9952894 IC50 = 8800 nM T50773 CQ8J7T 9953181 IC50 = 54000 nM T50773 C8OX9T 9964212 IC50 = 730000 nM T50773 C8THS1 9970277 IC50 = 85 nM T50773 CT6XQ2 9983092 IC50 = 51000 nM T50773 C18ZXU 9990413 IC50 = 220 nM T50773 CVG9I2 10012350 IC50 = 1840 nM T50773 C4KT7I 10014539 IC50 = 69000 nM T50773 CV85MG 10019118 IC50 = 0.22 nM T50773 CSZ75E 10046311 IC50 = 21000 nM T50773 CRG1N0 10058240 IC50 = 130000 nM T50773 C64ZDU 10059633 IC50 = 1.8 nM T50773 CI1Q6X 10081481 IC50 = 450 nM T50773 CHC82B 10083376 IC50 = 48400 nM T50773 CSHQ57 10084828 IC50 = 52000 nM T50773 C06KTL 10087724 IC50 = 54.7 nM T50773 C83ZDL 10096130 IC50 = 1100 nM T50773 CKY4R8 10112957 Ki > 22385 nM T50773 C0Q7BK 10127057 IC50 > 100000 nM T50773 C9ERD7 10130575 IC50 = 86 nM T50773 CLZF79 10133903 Ki > 22385 nM T50773 C2RW5Z 10135822 Ki > 22385 nM T50773 C4U3IC 10144962 IC50 > 100000 nM T50773 C2H0UF 10149048 IC50 = 60 nM T50773 CUE7K0 10156677 Ki > 22385 nM T50773 CUB1G7 10157334 Ki > 22385 nM T50773 C6PZ1U 10160012 Ki > 22385 nM T50773 C0L1KV 10162433 Ki > 22385 nM T50773 C29RUO 10162817 Ki > 22385 nM T50773 C6S5OX 10179212 Ki = 3949 nM T50773 CF7C3M 10180260 Ki = 701 nM T50773 C4FC2O 10183667 IC50 > 100000 nM T50773 CWU9N2 10198228 IC50 = 770 nM T50773 C05DXJ 10200731 Ki > 22385 nM T50773 C6ISW4 10203198 Ki > 22385 nM T50773 CD2U3A 10203599 Ki = 1127 nM T50773 CQ8N1T 10209865 IC50 = 7700 nM T50773 CQ0V1C 10219838 IC50 = 9900 nM T50773 CBZ3P2 10221723 Ki = 14421 nM T50773 CBC45I 10222923 Ki > 22385 nM T50773 CZ92XV 10225547 Ki = 17258 nM T50773 CU9W8N 10233525 IC50 = 15000 nM T50773 C5P0AO 10238227 IC50 = 47000 nM T50773 CCS75T 10242745 IC50 = 177000 nM T50773 CZ90LD 10250452 IC50 = 24 nM T50773 CU8C5K 10254918 IC50 = 49000 nM T50773 C17HUN 10255762 IC50 = 46000 nM T50773 CQ07AR 10270647 Ki > 22385 nM T50773 CD0P5E 10271196 Ki > 22385 nM T50773 CQ36IM 10272290 Ki = 523 nM T50773 CA7Q8J 10298482 Ki = 1066 nM T50773 CY3LK8 10300368 Ki > 22385 nM T50773 C9FZ2O 10304081 IC50 > 100000 nM T50773 C8J3NA 10304145 IC50 = 450 nM T50773 C7US0V 10304855 IC50 = 66000 nM T50773 CJDY62 10306170 IC50 = 19000 nM T50773 C3FB4T 10310021 IC50 = 74000 nM T50773 CY6N9I 10318743 IC50 = 35000 nM T50773 C08UHI 10320529 IC50 > 1000000 nM T50773 CNV4R3 10324641 IC50 = 15000 nM T50773 CIAV18 10333629 IC50 = 12.5 nM T50773 CL72FC 10334538 IC50 = 42000 nM T50773 CXP16T 10340933 IC50 > 1000000 nM T50773 C1AEN6 10341846 IC50 > 500000 nM T50773 CEZ95L 10342016 IC50 = 9400 nM T50773 CKZT43 10353699 IC50 = 1.5 nM T50773 CW70CV 10376453 IC50 = 7.4 nM T50773 CK07VX 10376940 IC50 = 9900 nM T50773 CQ7J2Z 10383508 IC50 > 20000 nM T50773 CY5M4R 10388027 IC50 = 11000 nM T50773 CHZ85I 10393133 IC50 > 500000 nM T50773 CLI51Z 10398371 IC50 = 200 nM T50773 C8NAX7 10403949 IC50 = 0.55 nM T50773 CVK1G5 10412922 IC50 = 15000 nM T50773 C92DAJ 10415172 IC50 > 1000000 nM T50773 C1O2RY 10426457 IC50 > 100000 nM T50773 C80ZBS 10429788 IC50 > 100000 nM T50773 C6GHF1 10433039 IC50 = 39000 nM T50773 CWCA76 10439426 IC50 > 100000 nM T50773 CAF71Y 10443207 IC50 = 1600 nM T50773 CO59EL 10450114 IC50 = 59000 nM T50773 C4OC6P 10455620 IC50 = 23000 nM T50773 C1WKE4 10455621 IC50 > 100000 nM T50773 CHP37D 10456407 IC50 > 1000000 nM T50773 CLV58Q 10468265 IC50 = 17 nM T50773 CH1DG5 10478099 IC50 = 77000 nM T50773 CK3IW4 10584272 IC50 = 111000 nM T50773 C0KTQ5 10607253 IC50 = 730000 nM T50773 C4PJ7H 10656779 IC50 = 42000 nM T50773 CHA8X6 10751333 IC50 = 30000 nM T50773 CYLO09 10774283 IC50 = 52000 nM T50773 CL26WQ 10780092 IC50 = 49000 nM T50773 C2KDY6 10798619 IC50 = 228000 nM T50773 C1WG0P 10798659 IC50 = 38 nM T50773 C1ZJ4I 10799226 IC50 = 43000 nM T50773 CJKX61 10821833 IC50 = 59000 nM T50773 C7BLJ1 10821834 IC50 > 100000 nM T50773 C3E8ID 10845163 IC50 = 288000 nM T50773 CK9SB4 10845727 IC50 = 299000 nM T50773 CJ39DG 10872395 IC50 = 32900 nM T50773 CY9CW2 10969177 IC50 = 12000 nM T50773 CT75CX 10982631 IC50 > 125000 nM T50773 CZ94WH 11025199 IC50 = 40400 nM T50773 C4MD5V 11037154 IC50 > 1000000 nM T50773 CH4TD3 11037548 IC50 = 60000 nM T50773 C9S8AG 11068388 IC50 = 79000 nM T50773 C60JXQ 11079321 IC50 = 87300 nM T50773 COAR21 11101478 IC50 > 100000 nM T50773 C6QL3H 11122260 IC50 = 36100 nM T50773 C26ODF 11150893 IC50 = 185 nM T50773 CSB2T9 11166406 IC50 = 4.2 nM T50773 CO9QM2 11198569 IC50 > 100000 nM T50773 CF1LD8 11199808 Ki > 3000 nM T50773 C68XFD 11205761 IC50 > 1000000 nM T50773 C3BXS4 11206225 IC50 > 500000 nM T50773 CMBT59 11207320 IC50 = 7500 nM T50773 CW8FL2 11209569 IC50 = 1.31 nM T50773 CJB87Z 11210511 IC50 = 38000 nM T50773 C6VKT5 11219158 IC50 = 25500 nM T50773 CXAR72 11220471 IC50 = 1.77 nM T50773 CK1UE7 11229192 IC50 = 152000 nM T50773 C35JSU 11229576 IC50 = 38 nM T50773 C3X9SY 11229581 IC50 = 276000 nM T50773 CHX25W 11232123 IC50 = 5 nM T50773 C0JD5Q 11232605 IC50 = 1.1 nM T50773 CYL67P 11232890 Ki = 1545 nM T50773 C5AB7G 11236208 IC50 = 6800 nM T50773 C5CZH3 11242300 IC50 = 16300 nM T50773 CUS5G2 11243728 IC50 = 23.5 nM T50773 CH82RJ 11244267 IC50 = 113 nM T50773 CLJ7A1 11255193 IC50 = 0.66 nM T50773 C61KZW 11266019 IC50 = 1.1 nM T50773 CKL1A8 11268930 Ki = 2347 nM T50773 CM0YI7 11269397 Ki = 5460 nM T50773 C5IY0L 11269712 IC50 = 95000 nM T50773 CM1A5F 11270889 IC50 = 18000 nM T50773 CR46GY 11277009 IC50 = 63000 nM T50773 C0U2MV 11289193 IC50 = 4.6 nM T50773 CTC0P9 11289792 IC50 = 1.1 nM T50773 C51QAB 11300739 IC50 = 7.4 nM T50773 C2SOA8 11306467 IC50 = 78000 nM T50773 C06NLF 11309656 IC50 = 65000 nM T50773 C8I1QE 11310450 IC50 = 48000 nM T50773 C47GSV 11310499 IC50 = 2900 nM T50773 CP9LQ0 11312069 IC50 = 0.8 nM T50773 C4GUX3 11312733 IC50 = 1.91 nM T50773 CEZ27P 11314348 Ki = 1943 nM T50773 CTG12Q 11321743 IC50 = 1200 nM T50773 C38ADT 11346439 IC50 = 0.75 nM T50773 C5SR4K 11346707 IC50 = 133500 nM T50773 CNB7G8 11356095 IC50 = 9900 nM T50773 C24QLP 11356421 IC50 = 500000 nM T50773 C1WOH9 11359214 IC50 = 2.3 nM T50773 CKP0G9 11362130 IC50 = 17000 nM T50773 CZ37IN 11372458 IC50 = 0.41 nM T50773 CW3QZ7 11374531 IC50 > 100000 nM T50773 C30JEU 11381416 IC50 > 30000 nM T50773 C9FN7U 11381726 IC50 = 1.13 nM T50773 CH74XT 11383468 IC50 = 0.39 nM T50773 CML13R 11389441 IC50 = 179000 nM T50773 CL9HN3 11395030 Ki > 3000 nM T50773 CSR53F 11404106 IC50 = 1.34 nM T50773 CTW02K 11406276 Ki > 3000 nM T50773 C0RIS4 11417008 IC50 = 21000 nM T50773 CRZ5F1 11418876 IC50 > 100000 nM T50773 CY15PU 11429829 Ki = 417 nM T50773 C27ITV 11436930 IC50 = 1.5 nM T50773 CLF89Y 11437087 IC50 = 18.6 nM T50773 CH39KX 11437726 IC50 = 0.9 nM T50773 CH09SE 11447824 IC50 = 4900 nM T50773 CUG51Q 11449442 IC50 = 2.7 nM T50773 C9RZC1 11450265 IC50 = 0.39 nM T50773 CW27UK 11450266 IC50 = 0.62 nM T50773 C7TOQ4 11472776 IC50 = 187 nM T50773 CO7T4W 11473127 IC50 = 2.7 nM T50773 C53RWU 11474019 IC50 = 0.6 nM T50773 CE5A4M 11475797 IC50 = 42000 nM T50773 C7JWD3 11476287 IC50 > 100000 nM T50773 CS4H7X 11481506 IC50 = 577 nM T50773 CTD0S4 11486251 Ki > 3000 nM T50773 CNMA97 11487118 IC50 = 98000 nM T50773 C06RUA 11493219 IC50 > 30000 nM T50773 C9PRY1 11494684 IC50 > 100000 nM T50773 CAH5Z6 11500899 IC50 > 30000 nM T50773 C15UQK 11515912 IC50 = 31248 nM T50773 C2TCM8 11523077 IC50 = 68000 nM T50773 CMYN65 11526865 IC50 > 100000 nM T50773 C0O3XD 11527019 IC50 = 17600 nM T50773 CZ35WN 11533932 IC50 > 100000 nM T50773 CKM89Z 11538673 IC50 = 31165 nM T50773 CMD6H8 11538715 IC50 = 8470 nM T50773 CG7I8Z 11538992 IC50 > 100000 nM T50773 CPR71X 11540951 IC50 > 100000 nM T50773 C98GDW 11541277 IC50 > 100000 nM T50773 CBR9K8 11541314 IC50 = 18000 nM T50773 CVT52Y 11545508 IC50 = 50146 nM T50773 CMN2K0 11566106 IC50 = 20720 nM T50773 CI5W4Y 11566450 IC50 > 30000 nM T50773 CY0A7J 11570138 IC50 > 100000 nM T50773 C6F4OE 11573417 IC50 > 100000 nM T50773 CAE39I 11573427 IC50 > 30000 nM T50773 CCR9Q2 11574031 IC50 = 36003 nM T50773 CQU80H 11576569 IC50 > 100000 nM T50773 CW94NS 11577331 IC50 > 100000 nM T50773 CQ86GI 11577431 IC50 > 100000 nM T50773 CVG3B6 11580945 IC50 > 100000 nM T50773 CCR0D7 11581247 IC50 > 100000 nM T50773 CYT4Z1 11581458 IC50 = 34201 nM T50773 CAZL49 11584650 IC50 > 100000 nM T50773 C5JYV7 11591936 IC50 = 63000 nM T50773 CSCW37 11592154 IC50 = 59000 nM T50773 C9MXO0 11596219 IC50 > 20000 nM T50773 CMUV42 11596607 IC50 = 2880 nM T50773 CPXV24 11603996 IC50 = 6400 nM T50773 CL4NM7 11604454 IC50 > 100000 nM T50773 C15DLO 11608317 IC50 = 0.48 nM T50773 CQL5S8 11613750 IC50 = 26000 nM T50773 CD3YU1 11616861 IC50 > 30000 nM T50773 CEX4O6 11617338 IC50 = 18869 nM T50773 C2APG7 11623550 IC50 > 30000 nM T50773 CDZ72J 11624893 IC50 > 20000 nM T50773 C7YKC0 11628195 IC50 > 100000 nM T50773 C3RZO9 11645337 IC50 = 17400 nM T50773 CXG1B4 11649741 IC50 = 61000 nM T50773 C3Y7EL 11678025 IC50 > 100000 nM T50773 CV0XW8 11680991 IC50 = 5717.6 nM T50773 CNF1M4 11681778 IC50 > 20000 nM T50773 C0IWC9 11689866 IC50 > 100000 nM T50773 C79ECL 11695535 IC50 > 100000 nM T50773 C8SI4E 11702902 IC50 > 20000 nM T50773 C0Q3IL 11703158 IC50 = 29315 nM T50773 CFO63Q 11704578 IC50 = 6452 nM T50773 CU8LZ4 11705859 IC50 > 10000 nM T50773 CCR80L 11717090 IC50 > 100000 nM T50773 CZS71R 11717268 IC50 = 34444 nM T50773 CIEJ54 11720809 IC50 = 14000 nM T50773 CHA7Z9 11722557 IC50 = 25380 nM T50773 CJ6XR8 11730284 IC50 = 3800 nM T50773 CX9U4G 11731880 IC50 > 1000000 nM T50773 C1P9ZM 11776124 IC50 = 397000 nM T50773 CO73AL 11784400 IC50 > 100000 nM T50773 C6ET2R 11817181 IC50 = 15700 nM T50773 CK24XY 11819467 IC50 = 1840 nM T50773 C19HAP 11825584 IC50 > 1000000 nM T50773 CQY50P 12742483 IC50 = 88700 nM T50773 CJAE28 15036410 IC50 = 9800 nM T50773 C6BHJ9 15101668 IC50 = 390000 nM T50773 C13JIX 15949418 IC50 > 100000 nM T50773 C49NUJ 15949507 IC50 = 61000 nM T50773 C8M0FT 15951543 IC50 = 4.1 nM T50773 CI3DB4 15951636 IC50 > 100000 nM T50773 C3SM4T 15951642 IC50 > 100000 nM T50773 CL1E6O 15953860 IC50 > 100000 nM T50773 C13-MAR 16040457 IC50 > 100000 nM T50773 C0YQ9A 16046127 IC50 = 0.62 nM T50773 CS7DQ3 16090844 Ki > 30000 nM T50773 C8CVG9 16090856 Ki > 30000 nM T50773 CA1PV5 16216352 IC50 = 0.88 nM T50773 CD9MQ6 16223559 IC50 > 20000 nM T50773 CQ7G8T 16223560 IC50 > 20000 nM T50773 CN24YP 16223762 IC50 > 20000 nM T50773 CF37TH 16226604 IC50 > 20000 nM T50773 C6ANU2 16226605 IC50 > 20000 nM T50773 CT01PQ 16739331 IC50 = 18190 nM T50773 C61RFP 16755651 IC50 = 4130 nM T50773 C15TBF 17751406 IC50 = 16520 nM T50773 CX5F2U 17763521 IC50 > 500000 nM T50773 CV4Z6Q 18398587 IC50 = 2100 nM T50773 CP3S0V 18398588 IC50 = 1600 nM T50773 CC8RN3 20198196 IC50 = 630 nM T50773 CBZ1E6 21045424 IC50 = 44000 nM T50773 CPES59 21949259 IC50 = 65000 nM T50773 C2W4KV 21949272 IC50 = 62000 nM T50773 C0X4SO 22029457 IC50 > 100000 nM T50773 CLK4G6 22029894 IC50 > 100000 nM T50773 CED47V 22690988 IC50 = 122000 nM T50773 C9VGC8 22691359 IC50 > 100000 nM T50773 C1M2ZS 22691666 IC50 > 100000 nM T50773 CM4SH2 23595882 IC50 > 500000 nM T50773 C8JSI4 23628284 IC50 = 72000 nM T50773 CAQ81M 23644660 IC50 > 100000 nM T50773 CDPU25 23644665 IC50 = 2500 nM T50773 CCSU21 23645371 IC50 = 84430 nM T50773 CFV07G 23645410 IC50 = 64000 nM T50773 CIMG82 23645411 IC50 > 100000 nM T50773 C2Q5IK 23645581 IC50 = 12000 nM T50773 CP9GS5 23645686 IC50 = 5700 nM T50773 C6R2LP 23645687 IC50 = 1000 nM T50773 CN7FK3 23645688 IC50 = 2500 nM T50773 CSHX17 23645689 IC50 = 4500 nM T50773 CL8QV6 23645690 IC50 = 1800 nM T50773 C0AU9X 23645691 IC50 = 2200 nM T50773 CRM3Y4 23645692 IC50 = 4300 nM T50773 CDM8A2 23645693 IC50 = 3800 nM T50773 CIR1F6 23645694 IC50 = 5200 nM T50773 CK5G6I 23645695 IC50 = 6000 nM T50773 CHS76O 23645696 IC50 = 24400 nM T50773 CVP59D 23645697 IC50 = 26800 nM T50773 CH13BW 23645698 IC50 = 15000 nM T50773 CL0K1T 23645699 IC50 = 5400 nM T50773 CB3Z7O 23645700 IC50 = 8100 nM T50773 CNO6Q1 23645702 IC50 = 1300 nM T50773 CGMC54 23645703 IC50 = 3000 nM T50773 C0V4WR 23645705 IC50 = 14100 nM T50773 CKM6Y8 23645917 IC50 = 71000 nM T50773 C9Y2ZL 23645918 IC50 = 71000 nM T50773 C4V6BX 23645919 IC50 = 38000 nM T50773 C78PNU 23645920 IC50 = 51000 nM T50773 C5YT6S 23645921 IC50 = 16000 nM T50773 CELQ89 23645922 IC50 = 18000 nM T50773 CGV92H 23645923 IC50 = 17000 nM T50773 CJ60EH 23645924 IC50 = 5500 nM T50773 CZG70A 23645925 IC50 = 67000 nM T50773 CD6V7X 23645926 IC50 = 40000 nM T50773 C1TD4J 23645927 IC50 = 92000 nM T50773 C71PQU 23645928 IC50 = 43000 nM T50773 C8EOB9 23645929 IC50 = 26000 nM T50773 C0M1TH 23645930 IC50 = 4000 nM T50773 CFHB36 23645931 IC50 = 54000 nM T50773 CTG27F 23645932 IC50 = 30000 nM T50773 CS2FT5 23645933 IC50 = 67000 nM T50773 C98QGK 23645934 IC50 = 43000 nM T50773 CS76DY 23645935 IC50 = 85000 nM T50773 C91MYK 23645936 IC50 > 100000 nM T50773 C3AQC0 23645937 IC50 = 31000 nM T50773 C61GTC 23645938 IC50 = 80000 nM T50773 C8XF6R 23645939 IC50 = 63000 nM T50773 C7IX5B 23645940 IC50 = 15000 nM T50773 CP6M3W 23645941 IC50 = 11000 nM T50773 CQ75XK 23645942 IC50 = 1900 nM T50773 C8T7GY 23645943 IC50 = 35000 nM T50773 C25ZXC 23645944 IC50 = 56000 nM T50773 C4A3NI 23645945 IC50 > 100000 nM T50773 C9Y1BP 23646016 IC50 > 20000 nM T50773 CL8DY2 23646017 IC50 > 20000 nM T50773 CT6Q1R 23646018 IC50 > 20000 nM T50773 C8VS1X 23646019 IC50 > 20000 nM T50773 CL4BX5 23646020 IC50 > 20000 nM T50773 CZ24WC 23646021 IC50 > 20000 nM T50773 C98VYW 23646022 IC50 > 20000 nM T50773 CCL17M 23646023 IC50 > 20000 nM T50773 CT16HE 23646024 IC50 = 19250 nM T50773 CAL8T5 23646025 IC50 = 31259 nM T50773 CVSH12 23646026 IC50 > 100000 nM T50773 C15HJB 23646027 IC50 > 100000 nM T50773 CBUM54 23646029 IC50 > 100000 nM T50773 C32ZNH 23646030 IC50 = 27537 nM T50773 CE8L2I 23646031 IC50 = 19000 nM T50773 C8SIU2 23646032 IC50 = 20891 nM T50773 C7L6JR 23646033 IC50 > 100000 nM T50773 CJ9ZL3 23646080 IC50 = 90000 nM T50773 C0S2UB 23646081 IC50 = 37800 nM T50773 CQ3KF6 23646082 IC50 = 15500 nM T50773 CZ9P0Q 23646083 IC50 = 10800 nM T50773 CFPN10 23646084 IC50 = 15700 nM T50773 C0NV1B 23646085 IC50 = 27200 nM T50773 CSW9T1 23646086 IC50 = 1300 nM T50773 CH72RP 23646087 IC50 = 53700 nM T50773 CH5Y2F 23646088 IC50 = 500000 nM T50773 CJ47OR 23646089 IC50 = 91300 nM T50773 CRT2B0 23646090 IC50 = 100000 nM T50773 C7JXN0 23646091 IC50 = 34000 nM T50773 C4K1NE 23646092 IC50 = 13400 nM T50773 CJV2K1 23646093 IC50 = 12900 nM T50773 C51BSR 23646094 IC50 = 21900 nM T50773 C2WDG4 23646095 IC50 = 9600 nM T50773 CB2ZT7 23646096 IC50 = 11000 nM T50773 COF57U 23646097 IC50 = 4200 nM T50773 CU26YP 23646098 IC50 = 1040 nM T50773 CM37ZS 23646100 IC50 = 54600 nM T50773 C4SV2J 23646101 IC50 = 62000 nM T50773 CX68KV 23646102 IC50 = 26000 nM T50773 CUZ0D8 23646448 IC50 > 100000 nM T50773 C7PE0S 23646449 IC50 = 47000 nM T50773 COT87G 23646450 IC50 = 17000 nM T50773 CF2J9Q 23646451 IC50 = 89000 nM T50773 CFOA63 23647106 IC50 = 18000 nM T50773 CFTW63 23647114 IC50 > 100000 nM T50773 C0BQ2D 23647115 IC50 > 100000 nM T50773 CLO1Y2 23647116 IC50 > 100000 nM T50773 CSJ78F 23647117 IC50 > 100000 nM T50773 CDE9L7 23647118 IC50 > 100000 nM T50773 CZF25M 23647119 IC50 = 78000 nM T50773 CW5U3C 23647120 IC50 = 17000 nM T50773 CWO62C 23647121 IC50 = 56000 nM T50773 C0X1CK 23647122 IC50 = 22000 nM T50773 C7JOV9 23647123 IC50 = 71000 nM T50773 C0UT7J 23647124 IC50 = 73000 nM T50773 C8P2VJ 23647125 IC50 = 61000 nM T50773 CQ85KB 23647126 IC50 = 90000 nM T50773 CRFL12 23647127 IC50 = 31000 nM T50773 CP3CF0 23647128 IC50 = 42000 nM T50773 CJA3M7 23647129 IC50 = 17000 nM T50773 C7L3RX 23647130 IC50 = 27000 nM T50773 C8UWB7 23647132 IC50 = 49000 nM T50773 C60MWC 23647133 IC50 = 8700 nM T50773 CO9GD8 23655077 IC50 = 145800 nM T50773 CPCX60 23655474 IC50 > 250000 nM T50773 CB1E5P 23655476 IC50 > 1000000 nM T50773 CWTD09 23655478 IC50 > 1000000 nM T50773 CW9UR3 23657402 IC50 > 250000 nM T50773 CU18EA 23657547 IC50 > 100000 nM T50773 CVF6E2 23661697 IC50 = 25000 nM T50773 CM7C4W 23661708 IC50 > 100000 nM T50773 CO6L9F 23661716 IC50 > 100000 nM T50773 CHR14F 23661718 IC50 = 74000 nM T50773 CNP9T1 24180585 IC50 = 19000 nM T50773 CO0ZA3 24692381 IC50 = 62000 nM T50773 CR7I3Y 24703639 IC50 = 500000 nM T50773 CVA72K 24704198 IC50 = 228000 nM T50773 CKWZ51 24710701 IC50 > 1000000 nM T50773 CU7W4F 24768547 IC50 = 130 nM T50773 CX8DH1 24769723 IC50 = 34000 nM T50773 C0H8OB 24776705 IC50 = 39000 nM T50773 C24GLZ 24776939 IC50 = 33000 nM T50773 C6LD2J 24777439 IC50 > 100000 nM T50773 CK8EL5 24777568 IC50 > 100000 nM T50773 CQ20PV 24777692 IC50 > 100000 nM T50773 C1WF3I 24777804 IC50 > 100000 nM T50773 C29SZR 24784416 IC50 = 29000 nM T50773 C8FQT4 24784664 IC50 > 100000 nM T50773 C2KL7G 24794725 IC50 = 31259 nM T50773 CKZ25G 24862861 IC50 = 330 nM T50773 CMK9B7 24894026 IC50 = 21500 nM T50773 CSIK84 24906298 IC50 = 191000 nM T50773 C7IDX9 25132160 IC50 = 160 nM T50773 CSU0B5 25189891 Ki > 30000 nM T50773 C7KN2U 42608447 IC50 = 8100 nM T50773 C60SVD 42636924 IC50 > 20000 nM T50773 C76NLT 42773972 IC50 = 14400 nM T50773 C6LQN3 43181622 IC50 = 136000 nM T50773 C42OZD 43271345 IC50 = 213000 nM T50773 CK54OM 43650152 IC50 = 57100 nM T50773 CS40ML 44123747 IC50 > 50000 nM T50773 CSX10M 44138030 IC50 = 16800 nM T50773 C50EKW 44250174 IC50 = 3400 nM T50773 CRZI12 44266022 IC50 > 100000 nM T50773 CL3Q2J 44306072 IC50 = 18000 nM T50773 C2RC9I 44328126 IC50 = 150000 nM T50773 CTC40N 44328274 Ki = 1430 nM T50773 C8M0SH 44328300 IC50 = 110000 nM T50773 C6NZ9C 44328318 IC50 = 328 nM T50773 C6OHV2 44328319 IC50 > 500000 nM T50773 CA53DN 44330624 IC50 = 6.5 nM T50773 C7E1BJ 44330636 IC50 = 4 nM T50773 C75JRD 44360575 IC50 = 820 nM T50773 CS72FI 44360697 IC50 = 2000 nM T50773 CKSO92 44360724 IC50 = 12000 nM T50773 CYED53 44360725 IC50 = 6400 nM T50773 CXEC92 44360726 IC50 = 380 nM T50773 CL7WM8 44360734 IC50 = 4500 nM T50773 CA0U8X 44360744 IC50 = 8200 nM T50773 C50NME 44360749 IC50 = 4100 nM T50773 CKI6W3 44360785 IC50 = 170 nM T50773 CRM9Y7 44360786 IC50 = 960 nM T50773 CXTP74 44360787 IC50 = 15000 nM T50773 C5MB1D 44360809 IC50 = 8600 nM T50773 C29DTA 44360810 IC50 = 5000 nM T50773 C3M8KF 44360910 IC50 = 230 nM T50773 CR7Q9N 44360911 IC50 = 690 nM T50773 CFY7P3 44360924 IC50 = 360 nM T50773 C62HNE 44360925 IC50 = 340 nM T50773 C1H5YG 44360938 IC50 = 230 nM T50773 C6IZ8L 44360955 IC50 = 900 nM T50773 CCJA09 44360967 IC50 = 170 nM T50773 CLMF32 44360976 IC50 = 200 nM T50773 CV1YL5 44360977 IC50 = 170 nM T50773 CY8A9K 44361010 IC50 = 210 nM T50773 C2KWI0 44361074 IC50 = 170 nM T50773 C1Z2FV 44361086 IC50 = 350 nM T50773 C8MJY5 44361216 IC50 = 230 nM T50773 CYK42S 44361230 IC50 = 900 nM T50773 CM3R2T 44364102 IC50 = 32400 nM T50773 CJ0VM6 44364126 IC50 = 111000 nM T50773 C83IUZ 44364133 IC50 = 9900 nM T50773 CJ8N0S 44364172 IC50 = 78100 nM T50773 C7D2FW 44364210 IC50 = 299000 nM T50773 C8HO2F 44364211 IC50 = 159000 nM T50773 C9IQG4 44364212 IC50 = 51900 nM T50773 C47NKP 44364213 IC50 = 52000 nM T50773 C6CYU9 44364227 IC50 > 500000 nM T50773 CHLV59 44364231 IC50 = 10900 nM T50773 CZF5N2 44364237 IC50 = 490 nM T50773 C7VR0N 44364252 IC50 = 29300 nM T50773 CTS8U3 44364253 IC50 = 510 nM T50773 C0IW9L 44364296 IC50 = 140 nM T50773 C6FBH7 44364297 IC50 = 750 nM T50773 C79JMS 44364298 IC50 = 3000 nM T50773 C45IPD 44364338 IC50 = 288000 nM T50773 CF2TA0 44364385 IC50 = 38 nM T50773 C19DCN 44364405 IC50 = 1500 nM T50773 CX5AK7 44364446 IC50 = 158000 nM T50773 C4XIV2 44364456 IC50 = 4900 nM T50773 C3XN5A 44364457 IC50 = 43000 nM T50773 CKA86J 44364458 IC50 = 48000 nM T50773 CX8I6C 44381633 IC50 = 750 nM T50773 CW9F3N 44381634 IC50 = 540 nM T50773 CI39RJ 44381635 IC50 = 75 nM T50773 CLK90J 44381645 IC50 = 2000 nM T50773 CT0EO4 44381646 IC50 = 43 nM T50773 CHX2T7 44381647 IC50 = 630 nM T50773 C6Y4QW 44381687 IC50 = 5000 nM T50773 CN96MI 44381721 IC50 = 440 nM T50773 CK4SP1 44381763 IC50 = 780 nM T50773 CI6RT5 44381811 IC50 = 50000 nM T50773 CG1CD7 44381826 IC50 = 820 nM T50773 CL51SX 44381845 IC50 = 160 nM T50773 CXBY42 44381846 IC50 = 990 nM T50773 C5SV9U 44381847 IC50 = 270 nM T50773 CRY5K1 44381848 IC50 = 870 nM T50773 CRE8J7 44381849 IC50 = 14 nM T50773 CUX2Q9 44381861 IC50 = 110 nM T50773 C92CKY 44381862 IC50 = 19000 nM T50773 CIX09S 44381884 IC50 = 2300 nM T50773 C3GH0S 44381896 IC50 = 26 nM T50773 C0FQO1 44381899 IC50 = 240 nM T50773 CTRX81 44381910 IC50 = 4000 nM T50773 C2XBA5 44381911 IC50 = 1700 nM T50773 CBL60E 44381919 IC50 = 3100 nM T50773 CARK25 44381928 IC50 = 430 nM T50773 C4LR3K 44381945 IC50 = 1400 nM T50773 CQ4VZ3 44381966 IC50 = 1300 nM T50773 CDCY49 44381967 IC50 = 250 nM T50773 CT9IN5 44381974 IC50 = 110 nM T50773 C0FQY4 44381979 IC50 = 260 nM T50773 CP7XG9 44382005 IC50 = 2500 nM T50773 C6YFP9 44382006 IC50 = 62000 nM T50773 CWJ3V5 44382013 IC50 = 110 nM T50773 CI8O3F 44382065 IC50 = 1000 nM T50773 CX2JS7 44382077 IC50 = 12000 nM T50773 C38MSH 44382133 IC50 = 53 nM T50773 C8PD7J 44382134 IC50 = 22 nM T50773 C89LXF 44382393 IC50 = 46000 nM T50773 CAJ50V 44382443 IC50 = 40000 nM T50773 C8ZP1A 44382444 IC50 = 420 nM T50773 CKOD04 44382521 IC50 = 220 nM T50773 CY2C8J 44387751 IC50 = 3100 nM T50773 CXSU53 44387755 IC50 = 92000 nM T50773 CALG81 44387756 IC50 > 250000 nM T50773 CL1M7V 44387758 IC50 = 12800 nM T50773 C6T2MW 44387765 IC50 = 67000 nM T50773 CA7KI2 44390794 IC50 > 100000 nM T50773 C7N1GB 44393611 IC50 > 100000 nM T50773 C08BMZ 44394001 IC50 = 65000 nM T50773 C3KH1Q 44394024 IC50 = 56050 nM T50773 C4QE5X 44394028 IC50 > 100000 nM T50773 CPF49E 44394029 IC50 > 100000 nM T50773 CS35UP 44394072 IC50 = 48510 nM T50773 CW79MD 44394073 IC50 = 78000 nM T50773 CW81MP 44394103 IC50 = 77560 nM T50773 C25SDY 44394118 IC50 = 26000 nM T50773 CU85FA 44394119 IC50 = 640 nM T50773 CJ18AZ 44394135 IC50 = 19000 nM T50773 CTEP50 44394136 IC50 = 15000 nM T50773 C4BO3S 44394155 IC50 = 13000 nM T50773 C4B9OH 44394173 IC50 = 280 nM T50773 C85SEO 44394194 IC50 > 100000 nM T50773 CS1Z7X 44394195 IC50 = 82120 nM T50773 C39LZT 44394203 IC50 = 36190 nM T50773 CF6Y8L 44394209 IC50 = 5775 nM T50773 CQ09FB 44394210 IC50 > 100000 nM T50773 CXG8B6 44394238 IC50 = 49700 nM T50773 CIJ95E 44394239 IC50 = 92060 nM T50773 C3Q5WZ 44394241 IC50 = 24570 nM T50773 CL3EP4 44394242 IC50 = 12000 nM T50773 C8U2ZQ 44394244 IC50 = 67630 nM T50773 CZA46H 44394270 IC50 = 48510 nM T50773 CUGH58 44394271 IC50 = 29750 nM T50773 CG53YO 44394349 IC50 = 24330 nM T50773 C59NLA 44394350 IC50 = 33890 nM T50773 CPX1M9 44403336 IC50 = 18 nM T50773 CSEN70 44403337 IC50 = 40 nM T50773 C0NXE8 44403338 IC50 = 8.2 nM T50773 C91MNA 44403353 IC50 = 0.48 nM T50773 CR53EK 44403354 IC50 = 4.7 nM T50773 C8MLN6 44403355 IC50 = 3.7 nM T50773 CBAZ94 44403359 IC50 = 890 nM T50773 CRO16Q 44403360 IC50 = 2 nM T50773 C0FC7D 44403361 IC50 = 0.72 nM T50773 CGYM03 44403370 IC50 = 5500 nM T50773 C26QCP 44403378 IC50 = 2600 nM T50773 CTZ25G 44403379 IC50 = 130 nM T50773 C3HFZ7 44403391 IC50 = 570 nM T50773 C3TOY4 44403392 IC50 = 140 nM T50773 CU39LX 44403393 IC50 = 15 nM T50773 CIA8Y3 44403397 IC50 = 4 nM T50773 C6P7NE 44403398 IC50 = 2.2 nM T50773 CP34SF 44403405 IC50 = 420 nM T50773 C60VBT 44403406 IC50 = 1 nM T50773 CQ5T4Y 44403412 IC50 = 6.3 nM T50773 CMX9B1 44403416 IC50 = 120 nM T50773 CUKG07 44403417 IC50 = 35 nM T50773 CX29FU 44403421 IC50 = 4600 nM T50773 C2P4CQ 44403422 IC50 = 1.8 nM T50773 C41IAB 44403437 IC50 = 220 nM T50773 CCOA39 44403438 IC50 = 49 nM T50773 CLYJ80 44403439 IC50 = 71 nM T50773 C4YAH3 44404393 IC50 = 8 nM T50773 C02SYC 44406179 Ki > 22385 nM T50773 CU8B3S 44406189 Ki > 22385 nM T50773 C5P1RX 44406284 Ki > 22385 nM T50773 CGJ17L 44415883 IC50 = 57 nM T50773 CE0KW2 44415905 IC50 = 3.4 nM T50773 CPR49A 44415906 IC50 = 19 nM T50773 CQ5P2J 44415929 IC50 = 84 nM T50773 CM2W5X 44415930 IC50 = 3.8 nM T50773 COPZ87 44415944 IC50 = 46.5 nM T50773 CE7UB0 44418114 IC50 = 75000 nM T50773 C70KAO 44418211 IC50 > 20000 nM T50773 C8LC2A 44418213 IC50 > 20000 nM T50773 CTM1Y8 44418214 IC50 = 800 nM T50773 C1EMA5 44418215 IC50 > 20000 nM T50773 CWDH12 44418216 IC50 > 20000 nM T50773 C1FB4K 44418218 IC50 > 20000 nM T50773 CVC3R4 44418219 IC50 > 20000 nM T50773 CU1FG2 44418222 IC50 > 20000 nM T50773 C8ZH5R 44418223 IC50 > 20000 nM T50773 CA9YM3 44418225 IC50 > 20000 nM T50773 CQE5Y0 44418229 IC50 > 20000 nM T50773 C2LXS7 44418232 IC50 > 20000 nM T50773 C59HZQ 44418251 IC50 > 100000 nM T50773 C2UR9X 44418256 IC50 > 20000 nM T50773 CK20CA 44418257 IC50 > 20000 nM T50773 CO3GL6 44418260 IC50 > 20000 nM T50773 CY3O7C 44418261 IC50 > 20000 nM T50773 C0ITV9 44418262 IC50 > 20000 nM T50773 C68SHD 44418264 IC50 > 20000 nM T50773 CDI98V 44418265 IC50 > 20000 nM T50773 CHO5P1 44418266 IC50 > 20000 nM T50773 C95XQC 44418268 IC50 > 20000 nM T50773 CZ2MB8 44426068 IC50 = 59000 nM T50773 C8PKO5 44426070 IC50 > 100000 nM T50773 CR0A1M 44431316 IC50 > 100000 nM T50773 CV1R7A 44431317 IC50 > 100000 nM T50773 CY76AB 44432858 IC50 = 5470 nM T50773 CS95EU 44432859 IC50 = 70100 nM T50773 C1PX9V 44432860 IC50 = 10000 nM T50773 CE4Q5X 44432862 IC50 = 200 nM T50773 CHN6E3 44432863 IC50 = 35100 nM T50773 CF2AT6 44432881 IC50 < 390 nM T50773 CTD24F 44432889 IC50 < 390 nM T50773 CU67PL 44432901 IC50 = 3240 nM T50773 C35GZP 44432904 IC50 = 2070 nM T50773 C21UQD 44432911 IC50 = 2670 nM T50773 CU27DF 44432914 IC50 = 1250 nM T50773 C9E1SZ 44432915 IC50 = 10000 nM T50773 CZ47KB 44432929 IC50 = 97200 nM T50773 CS5BT9 44432935 IC50 > 10000 nM T50773 CI9M8R 44432936 IC50 < 390 nM T50773 C5LTR0 44432937 IC50 < 390 nM T50773 C6EJB0 44432938 IC50 = 8660 nM T50773 CJ7YN0 44432940 IC50 = 1380 nM T50773 CVZ3I2 44432942 IC50 = 60000 nM T50773 CT29BC 44432944 IC50 = 1710 nM T50773 CQDS95 44433224 IC50 = 15000 nM T50773 CE92DA 44435310 IC50 = 20000 nM T50773 C3SBK5 44435313 IC50 = 85000 nM T50773 CX7UN0 44435314 IC50 = 77000 nM T50773 CE7XI5 44435315 IC50 = 2200 nM T50773 CGAR49 44435316 IC50 > 250000 nM T50773 CA0NZ7 44443707 IC50 > 100000 nM T50773 C24ZHB 44443708 IC50 = 92000 nM T50773 C8R4OD 44443709 IC50 = 80000 nM T50773 CLDN63 44443710 IC50 > 100000 nM T50773 C7LNP2 44443711 IC50 = 76000 nM T50773 CJX2M7 44443712 IC50 = 49000 nM T50773 C6RST0 44443713 IC50 = 85000 nM T50773 C3YL9X 44443714 IC50 = 64000 nM T50773 CRH8M1 44443715 IC50 = 56000 nM T50773 CIB50E 44443717 IC50 = 33000 nM T50773 CK6QF4 44443719 IC50 = 58000 nM T50773 CX6O1P 44443720 IC50 > 100000 nM T50773 C0YV2D 44443723 IC50 = 45000 nM T50773 C1BUJ5 44443725 IC50 = 28000 nM T50773 CXS34I 44443727 IC50 = 76000 nM T50773 CCHS17 44443729 IC50 = 37000 nM T50773 C39KZG 44443736 IC50 = 30000 nM T50773 C5H8EJ 44443737 IC50 = 19000 nM T50773 CS3Y1G 44444344 IC50 > 100000 nM T50773 CL2U9C 44444352 IC50 = 4000 nM T50773 C8VE5T 44444353 IC50 = 72000 nM T50773 C8F5HC 44444371 IC50 = 60000 nM T50773 CEW50M 44444373 IC50 = 15000 nM T50773 CO0M7Y 44444375 IC50 = 7400 nM T50773 CS93BI 44444377 IC50 = 33000 nM T50773 C9J4FB 44444379 IC50 = 18000 nM T50773 C3YA4K 44444383 IC50 = 4100 nM T50773 C75OIP 44444386 IC50 = 26000 nM T50773 C4J6ZG 44444390 IC50 = 9600 nM T50773 C05EBU 44444391 IC50 = 22000 nM T50773 CSN27E 44445042 IC50 = 30000 nM T50773 CGN61Q 44445047 IC50 = 62000 nM T50773 CYW8E3 44445051 IC50 > 100000 nM T50773 CRG64M 44445053 IC50 = 52000 nM T50773 C6ZID3 44445055 IC50 = 57000 nM T50773 C72KOR 44445057 IC50 = 83000 nM T50773 C0RTA6 44445060 IC50 = 47000 nM T50773 CIK8G3 44445063 IC50 = 36000 nM T50773 CN05VX 44445065 IC50 > 100000 nM T50773 COA90R 44445067 IC50 > 100000 nM T50773 CVO9F2 44453648 IC50 = 330 nM T50773 C91FSI 44453672 IC50 = 3910 nM T50773 C5UET4 44453690 IC50 = 140 nM T50773 C2JE8C 44453692 IC50 = 250 nM T50773 C6EC4J 44453922 IC50 = 210 nM T50773 C4C6NK 44453968 IC50 = 1400 nM T50773 CDS52W 44453970 IC50 = 1160 nM T50773 C9V2HU 44454016 IC50 = 420 nM T50773 CHKT64 44458509 IC50 = 3000 nM T50773 CXWQ16 44458510 IC50 = 3200 nM T50773 CBSZ02 44458521 IC50 = 3500 nM T50773 CIA6J1 44458523 IC50 = 5200 nM T50773 C6LKZ7 44458534 IC50 = 410 nM T50773 CR41OX 44458540 IC50 = 7500 nM T50773 CNK09O 44458542 IC50 = 1100 nM T50773 CM65HC 44458548 IC50 = 600 nM T50773 CKM0F5 44458549 IC50 = 12000 nM T50773 CR4CP3 44458554 IC50 = 810 nM T50773 CU68KW 44458566 IC50 = 6100 nM T50773 CC7I6Y 44458573 IC50 = 4500 nM T50773 CCI52U 44458574 IC50 = 21000 nM T50773 C0K7EZ 44458575 IC50 = 25000 nM T50773 CNK64C 44458581 IC50 = 8100 nM T50773 CF7I9V 44458586 IC50 = 2000 nM T50773 CW7QX0 44458587 IC50 = 660 nM T50773 CJ7Y6A 44458592 IC50 = 8300 nM T50773 C9QMB2 44458594 IC50 = 20000 nM T50773 CPJW14 44458603 IC50 = 38000 nM T50773 C0K2SV 44458617 IC50 = 1900 nM T50773 CSIL15 44458629 IC50 = 5000 nM T50773 C3EZ1V 44458770 IC50 = 2800 nM T50773 C91DWY 44560396 IC50 = 12200 nM T50773 CZ9WJ0 44560397 IC50 > 100000 nM T50773 C0FLU7 44560398 IC50 = 23000 nM T50773 CX9BK6 44560399 IC50 = 68 nM T50773 CZ43JR 44560454 IC50 > 100000 nM T50773 CY38QP 44560549 IC50 > 100000 nM T50773 C7IL3K 44560550 IC50 = 13000 nM T50773 CF9J7Z 44560551 IC50 = 7400 nM T50773 C1QAI4 44560552 IC50 = 2600 nM T50773 CK25CG 44560553 IC50 = 66000 nM T50773 C4C9NG 44560554 IC50 > 50000 nM T50773 CKIH45 44560555 IC50 > 100000 nM T50773 C2LW3C 44560595 IC50 = 7100 nM T50773 C47WCK 44560596 IC50 = 47000 nM T50773 CL8AE5 44560597 IC50 = 12600 nM T50773 C1YJ8C 44560648 IC50 = 117 nM T50773 CY6GU1 44560649 IC50 = 365 nM T50773 C12EYZ 44560650 IC50 = 316 nM T50773 C7LY9V 44560651 IC50 = 416 nM T50773 CG5CB2 44560698 IC50 = 3400 nM T50773 CR56BA 44560699 IC50 = 860 nM T50773 CIA45R 44560700 IC50 = 1700 nM T50773 CAK3U5 44560701 IC50 = 1300 nM T50773 CJE42H 44560746 IC50 > 100000 nM T50773 C5OW2C 44560747 IC50 = 41000 nM T50773 CM2GN5 44560748 IC50 = 3500 nM T50773 C5FSB4 44560749 IC50 = 4500 nM T50773 C5WEG1 44560750 IC50 = 380 nM T50773 CN0KO4 44560770 IC50 = 86 nM T50773 CZSO82 44560823 IC50 = 230000 nM T50773 C4IVD9 44560824 IC50 = 19000 nM T50773 C4L3VZ 44560825 IC50 = 5700 nM T50773 CHV7S1 44560826 IC50 = 3700 nM T50773 CE3NF4 44560849 IC50 = 3100 nM T50773 CT6P5E 44560850 IC50 = 860 nM T50773 CTH9P2 44560851 IC50 = 60000 nM T50773 CGZ48C 44560928 IC50 = 1500 nM T50773 C9EK8A 44560929 IC50 = 393000 nM T50773 CM68VD 44560930 IC50 = 1020 nM T50773 C4SMJ1 44560961 IC50 = 840 nM T50773 C2I3TR 44560962 IC50 = 38000 nM T50773 CGV49L 44560963 IC50 = 24000 nM T50773 CY0L1G 44560964 IC50 = 310 nM T50773 C7FST1 44560988 IC50 = 350 nM T50773 CGOM86 44560989 IC50 = 90000 nM T50773 C74ZNK 44560990 IC50 = 25 nM T50773 C95AUS 44560991 IC50 = 34 nM T50773 C1U4YQ 44565237 IC50 = 5200 nM T50773 CRK69O 44565238 IC50 > 20000 nM T50773 C6M2WD 44565239 IC50 > 20000 nM T50773 CTZ9L0 44565254 IC50 > 20000 nM T50773 CEMV93 44565274 IC50 > 20000 nM T50773 C5E6PQ 44565275 IC50 > 20000 nM T50773 CI93OK 44565276 IC50 > 20000 nM T50773 C2HRF1 44565277 IC50 > 20000 nM T50773 CFEC28 44565466 IC50 = 16000 nM T50773 C5MON6 44565467 IC50 > 20000 nM T50773 CGA4U6 44565488 IC50 > 20000 nM T50773 C1BZ3I 44565489 IC50 > 20000 nM T50773 CP3C5F 44565490 IC50 > 20000 nM T50773 CRU86T 44565491 IC50 > 20000 nM T50773 C3C2DL 44565492 IC50 > 20000 nM T50773 CJ2W1P 44565512 IC50 > 20000 nM T50773 C5Z9GW 44565513 IC50 > 20000 nM T50773 C3I0MO 44565514 IC50 > 20000 nM T50773 CI3J6Y 44565535 IC50 > 20000 nM T50773 CB90XZ 44565536 IC50 > 20000 nM T50773 C01SLH 44565537 IC50 > 20000 nM T50773 C8Y2LX 44565538 IC50 > 20000 nM T50773 CXD19F 44565539 IC50 = 17000 nM T50773 CFK92H 44565583 IC50 = 2460 nM T50773 CA0O7F 44565585 IC50 > 30000 nM T50773 CPZ7J3 44565844 IC50 = 1230 nM T50773 C9BGR3 44565845 IC50 = 2260 nM T50773 CR83QA 44565869 IC50 = 7120 nM T50773 C6K2WL 44565870 IC50 = 660 nM T50773 C3UL2E 44565871 IC50 = 660 nM T50773 C9SL5D 44565872 IC50 = 210 nM T50773 CZBX95 44565889 IC50 = 20400 nM T50773 C1TLY0 44565890 IC50 = 28300 nM T50773 CEO20N 44565891 IC50 = 31400 nM T50773 COA7X5 44565892 IC50 = 11100 nM T50773 CRO3D2 44567651 IC50 = 5100 nM T50773 CM95OD 44567652 IC50 = 5100 nM T50773 CX6WL5 44567653 IC50 = 10800 nM T50773 C4MP9D 44567654 IC50 = 8750 nM T50773 CV23FP 44567668 IC50 = 13050 nM T50773 CD4C7Y 44567710 IC50 = 4000 nM T50773 C4CUJ6 44567711 IC50 = 11000 nM T50773 CK1C7W 44567712 IC50 = 6420 nM T50773 CTK1I9 44567713 IC50 = 1340 nM T50773 CM50CU 44567747 IC50 = 2800 nM T50773 CNA0I9 44567918 IC50 = 18100 nM T50773 C6BXT0 44567919 IC50 = 2760 nM T50773 CJ85MG 44567920 IC50 = 1200 nM T50773 CUJD19 44567976 IC50 = 10900 nM T50773 C5YB6E 44567977 IC50 = 1000 nM T50773 CNF09E 44567978 IC50 = 907 nM T50773 C70WEI 44567979 IC50 = 1000 nM T50773 CW7NB6 44568016 IC50 = 9000 nM T50773 CY8Z3F 44568017 IC50 = 9880 nM T50773 CRM76D 44568018 IC50 = 21800 nM T50773 CCG83U 44568057 IC50 = 406 nM T50773 C8XW9A 44568058 IC50 = 96 nM T50773 CMQ7D5 44568097 IC50 = 1300 nM T50773 C1F9OL 44568098 IC50 = 1300 nM T50773 CUYK75 44568099 IC50 > 10000 nM T50773 CZ81XF 44568100 IC50 = 4330 nM T50773 C6GT0A 44568134 IC50 > 10000 nM T50773 C6IW5D 44568135 IC50 = 3900 nM T50773 C3PWD8 44568136 IC50 = 1800 nM T50773 C4NCA7 44568169 IC50 = 16500 nM T50773 C8TXH9 44568170 IC50 = 2200 nM T50773 C17PZX 44568171 IC50 = 11000 nM T50773 C7SCJ1 44568172 IC50 = 226 nM T50773 CZCU54 44571949 IC50 = 46.77 nM T50773 CJ96CO 44571951 IC50 = 99.43 nM T50773 C7E6IB 44572718 IC50 > 20000 nM T50773 CUH81Y 44572719 IC50 = 15000 nM T50773 CJHR19 44572720 IC50 = 2600 nM T50773 CG71OU 44572782 IC50 > 20000 nM T50773 C2DQ0C 44589933 IC50 = 28400 nM T50773 CUZ3P0 44589935 IC50 = 85200 nM T50773 CRN4U5 44590696 IC50 > 100000 nM T50773 CTC24F 44590734 IC50 = 420 nM T50773 C91FTW 44591848 IC50 > 30000 nM T50773 CY78PR 44591849 IC50 > 30000 nM T50773 CE2LW5 44591850 IC50 = 10800 nM T50773 C82YQS 44592509 IC50 = 11100000 nM T50773 CWJ2U0 44592510 IC50 = 10200000 nM T50773 CQI40A 44592511 IC50 = 9110000 nM T50773 CY8R3Q 44593399 IC50 = 43000 nM T50773 CP8YC3 44593408 IC50 = 1780 nM T50773 C4L6NS 44593409 IC50 = 2500 nM T50773 CI0FT1 44593463 IC50 > 20000 nM T50773 C65KPR 45101722 IC50 = 7200 nM T50773 CXYT36 45101723 IC50 = 2000 nM T50773 C2RNP7 45102670 IC50 = 16000 nM T50773 CGZD98 45265711 IC50 > 100000 nM T50773 CCO76A 45266134 IC50 = 1500 nM T50773 CU4C5P 45266135 IC50 = 89000 nM T50773 CLVM20 45266136 IC50 = 57000 nM T50773 C8H9GV 45267527 IC50 = 700 nM T50773 CP9B0W 45267530 IC50 = 530 nM T50773 C3GJK0 45267531 IC50 = 2300 nM T50773 CN38QU 45268229 IC50 = 11000 nM T50773 CEQ16V 45268233 IC50 = 19000 nM T50773 C0QB1V 45268417 IC50 = 1700 nM T50773 C2S9ZT 45268436 IC50 = 29000 nM T50773 CX8WC0 45269123 IC50 = 12000 nM T50773 C9HR0K 45269274 IC50 = 4800 nM T50773 CZ1N2O 45269275 IC50 = 4400 nM T50773 CIE21V 45269276 IC50 = 11000 nM T50773 CWT60M 45269971 IC50 = 6300 nM T50773 C8QJ7X 45270108 IC50 = 1200 nM T50773 CYWK62 45270115 IC50 = 5600 nM T50773 CGF7Z6 45270958 IC50 = 3800 nM T50773 CH5S8Y 45270959 IC50 = 5500 nM T50773 C5NH6Q 45271791 IC50 = 600 nM T50773 C8Z3DK 45271794 IC50 = 1400 nM T50773 CX62YA 45271796 IC50 = 6500 nM T50773 CZ8EO2 45271803 IC50 = 9400 nM T50773 CJ7Q9E 45271813 IC50 = 1300 nM T50773 CJI2R6 45272664 IC50 = 1900 nM T50773 C49BKQ 45272672 IC50 = 1700 nM T50773 CP36CT 45272682 IC50 = 7300 nM T50773 C8NL4U 45272683 IC50 = 5900 nM T50773 C6S0OC 45273404 IC50 = 10000 nM T50773 CYMR87 45273573 IC50 = 340 nM T50773 CFL87A 45273581 IC50 = 890 nM T50773 C2XB0P 45273589 IC50 = 3400 nM T50773 C28PRV 45273594 IC50 = 3900 nM T50773 CSX2T9 45273602 IC50 = 9100 nM T50773 CMP59Q 45273603 IC50 = 6000 nM T50773 C28ZXW 45487888 IC50 = 7000 nM T50773 C2N3IZ 45487894 IC50 = 4000 nM T50773 CP62TC 45487898 IC50 = 2200 nM T50773 CWQ1R9 45487903 IC50 = 2800 nM T50773 C8H1KY 45487904 IC50 = 5600 nM T50773 C6X7WJ 45487908 IC50 = 3200 nM T50773 C5OXM9 45487915 IC50 = 11000 nM T50773 CPJ19X 45487917 IC50 = 38000 nM T50773 CV2R7M 45487920 IC50 = 3800 nM T50773 C57JRG 45487921 IC50 = 10000 nM T50773 C4JD1P 45487922 IC50 = 36000 nM T50773 CPB85R 45487926 IC50 = 23000 nM T50773 CTY16E 45487930 IC50 = 3800 nM T50773 C4QTL9 45487931 IC50 = 17000 nM T50773 CG9V0L 45487940 IC50 = 14000 nM T50773 C5XTV1 45487945 IC50 = 886 nM T50773 C3VK4G 45487946 IC50 = 2300 nM T50773 C0SNL2 46209134 IC50 = 87000 nM T50773 CE9M5C 46209244 IC50 = 56000 nM T50773 CW60IG 46209246 IC50 = 88000 nM T50773 CDP7Q4 46870369 IC50 = 900 nM T50773 CAL9K6 46891534 IC50 > 100000 nM T50773 C4XTW7 46893990 IC50 > 100000 nM T50773 C9JKO5 46905992 IC50 = 460 nM T50773 C8DSG7 46916343 IC50 > 100000 nM T50773 C3RO8F 46916345 IC50 > 100000 nM T50773 CX07LJ 46916346 IC50 > 100000 nM T50773 CF94MW 46916347 IC50 > 100000 nM T50773 CH3F7O 46916384 IC50 > 100000 nM T50773 CM8W6E 46916385 IC50 > 100000 nM T50773 C6FA9Q 46916386 IC50 > 100000 nM T50773 CAW86J 46916387 IC50 > 100000 nM T50773 C63HBE 46916388 IC50 > 100000 nM T50773 CD1CZ7 46916389 IC50 > 100000 nM T50773 CH80LK 46916433 IC50 > 100000 nM T50773 CN4A3P 46916435 IC50 > 100000 nM T50773 CUQ86M 46917047 IC50 > 100000 nM T50773 CS5X9L 46917048 IC50 > 100000 nM T50773 CZP24U 46917049 IC50 = 400 nM T50773 CGMJ52 46938499 IC50 > 100000 nM T50773 C5RAS7 46938602 IC50 > 100000 nM T50773 C3B1LX 46938704 IC50 > 100000 nM T50773 C5TU1F 46938705 IC50 > 100000 nM T50773 CAGP83 46938706 IC50 > 100000 nM T50773 CP9V8Q 46938799 IC50 > 100000 nM T50773 CAB2H9 46938802 IC50 > 100000 nM T50773 C80RAT 47370344 IC50 > 100000 nM T50773 CZ7A9E 49796933 IC50 = 59000 nM T50773 C5RF0Y 49796938 IC50 > 100000 nM T50773 CE0C3Y 49796939 IC50 > 100000 nM T50773 CI4ZE6 49796940 IC50 > 100000 nM T50773 CBD8K2 49796942 IC50 > 100000 nM T50773 CI25XP 49796945 IC50 = 55000 nM T50773 C8WYA5 49796953 IC50 > 100000 nM T50773 CQH86V 49796955 IC50 > 100000 nM T50773 CBMV50 49796972 IC50 = 2700 nM T50773 C8IL0K 49796973 IC50 > 100000 nM T50773 CA90LB 49796974 IC50 = 2500 nM T50773 C07DHG 49796977 IC50 = 700 nM T50773 CAS2P4 49796982 IC50 = 21000 nM T50773 CG79KT 49796985 IC50 = 15000 nM T50773 C4D8RE 49796990 IC50 > 100000 nM T50773 CUKB68 49796994 IC50 = 38000 nM T50773 CUR9B0 49796995 IC50 = 5600 nM T50773 CWHO58 49796998 IC50 > 100000 nM T50773 CX74RG 49796999 IC50 = 45000 nM T50773 C20MAQ 49797000 IC50 = 15000 nM T50773 CD67OX 49797001 IC50 > 100000 nM T50773 C9LEF5 49797002 IC50 = 8500 nM T50773 CO2AX9 49797003 IC50 = 40000 nM T50773 CEM61W 49797006 IC50 = 77000 nM T50773 C7Y0JL 49797007 IC50 = 48000 nM T50773 CW45IK 49797008 IC50 > 100000 nM T50773 C79JUI 49797011 IC50 > 100000 nM T50773 CVAK94 49797012 IC50 = 9400 nM T50773 CUK5J1 49797013 IC50 = 57000 nM T50773 C4ZK5C 49797014 IC50 = 29000 nM T50773 C1PV8J 49797015 IC50 = 94000 nM T50773 C9YEU6 49797016 IC50 = 58000 nM T50773 CZD4S2 49797017 IC50 = 76000 nM T50773 CKY80F 49797018 IC50 > 100000 nM T50773 CS0D8Q 49797021 IC50 = 7100 nM T50773 C3GF4M 49797022 IC50 > 100000 nM T50773 C8XZT9 49797023 IC50 = 55000 nM T50773 C5H2AS 49797024 IC50 = 100000 nM T50773 C4P0VW 49797025 IC50 = 43000 nM T50773 CVY8M1 49797028 IC50 = 90000 nM T50773 CM59HB 49797029 IC50 = 75000 nM T50773 CH7Y1J 49797030 IC50 = 5300 nM T50773 CX18HI 49797031 IC50 = 44000 nM T50773 CUM28Z 49797035 IC50 > 100000 nM T50773 COS23G 49797036 IC50 = 26000 nM T50773 C2TSG6 49797038 IC50 = 11000 nM T50773 C7BI3W 49797039 IC50 = 81000 nM T50773 C71THK 49797040 IC50 = 5700 nM T50773 C0SG5O 49797041 IC50 = 28000 nM T50773 CM37VB 49797042 IC50 = 5900 nM T50773 C51NUG 49797043 IC50 = 5600 nM T50773 C65WXC 49797044 IC50 = 5200 nM T50773 CHTO37 49797045 IC50 = 48000 nM T50773 CA8R5K 49797046 IC50 = 7800 nM T50773 CLAR35 49797047 IC50 = 3600 nM T50773 C9OCZ3 49797048 IC50 > 100000 nM T50773 C49RUW 49797049 IC50 = 11000 nM T50773 C4EHT7 49797050 IC50 = 14000 nM T50773 CW6G5R 49797051 IC50 = 5200 nM T50773 CUK6G0 49797052 IC50 = 3000 nM T50773 CJ1FE2 49797053 IC50 = 23000 nM T50773 CKJO08 49797054 IC50 = 46000 nM T50773 C70KVU 49797055 IC50 = 36000 nM T50773 CP59BI 49797056 IC50 = 5900 nM T50773 CEDL61 49797057 IC50 = 14000 nM T50773 C5J2LV 49797058 IC50 = 59000 nM T50773 CEI20Q 49797059 IC50 = 19000 nM T50773 C7B5DY 49797060 IC50 = 2900 nM T50773 C5B1RM 49797061 IC50 = 1100 nM T50773 C40HJC 49797062 IC50 = 4600 nM T50773 CL3P4H 49797063 IC50 = 350 nM T50773 CPC76U 49797064 IC50 = 96 nM T50773 C5F4JN 49797065 IC50 = 10000 nM T50773 C86HND 49797066 IC50 = 330 nM T50773 C8E4XD 49797067 IC50 = 720 nM T50773 CHO1U0 49797068 IC50 = 820 nM T50773 CO1TW7 49797069 IC50 = 960 nM T50773 CAD6W1 49797071 IC50 = 830 nM T50773 CQYU80 49797072 IC50 = 3100 nM T50773 CEZ38H 49797073 IC50 = 4800 nM T50773 C0CEU7 49797074 IC50 = 3600 nM T50773 C72JXY 49797075 IC50 = 1300 nM T50773 COA41Q 49797076 IC50 = 670 nM T50773 CPQ3Z2 49797077 IC50 = 870 nM T50773 C1WI0D 49797078 IC50 = 2000 nM T50773 C4D8XP 49797079 IC50 = 1100 nM T50773 CQG4J6 49797080 IC50 = 2500 nM T50773 CKM9S4 49797081 IC50 = 490 nM T50773 C3JRW0 49797082 IC50 = 8600 nM T50773 C27IEB 49797083 IC50 = 1300 nM T50773 C0JUL3 49797084 IC50 = 2900 nM T50773 C85DOL 49797085 IC50 = 3800 nM T50773 CEGO30 49797086 IC50 = 2500 nM T50773 C2TC3I 49797087 IC50 = 120 nM T50773 C04JWY 49797088 IC50 = 2000 nM T50773 CA2U4Y 49797089 IC50 = 9200 nM T50773 CFT46J 49797090 IC50 = 2500 nM T50773 C35TFW 49797091 IC50 = 380 nM T50773 CRL7Z5 49797092 IC50 = 1800 nM T50773 CYU74X 49797093 IC50 = 1200 nM T50773 C2O3SG 49797094 IC50 = 250 nM T50773 CFL3O2 49797106 IC50 = 3900 nM T50773 CF4NR7 49797107 IC50 = 810 nM T50773 CV9QW6 49797108 IC50 = 16000 nM T50773 CJZA65 49797109 IC50 = 1100 nM T50773 CBS36X 49797110 IC50 > 100000 nM T50773 C0STP5 49797111 IC50 = 14000 nM T50773 C7KV5R 49797112 IC50 = 6200 nM T50773 CJPX53 49797113 IC50 = 9000 nM T50773 C2OI0Y 49797114 IC50 = 5000 nM T50773 CW20FJ 49797115 IC50 = 8000 nM T50773 C9P6VU 49797116 IC50 = 7100 nM T50773 C67SIA 49797117 IC50 = 6100 nM T50773 CCI8Y0 49797118 IC50 = 24000 nM T50773 CE10UF 49797119 IC50 = 4500 nM T50773 CLH0V3 49797120 IC50 = 8500 nM T50773 C2N8WX 49797121 IC50 = 550 nM T50773 CNCE06 49797122 IC50 = 5900 nM T50773 C76UAB 49797123 IC50 = 7400 nM T50773 CHWT89 49797124 IC50 = 2500 nM T50773 C1Z6NE 49797125 IC50 = 5500 nM T50773 C25MQG 49797126 IC50 = 2100 nM T50773 COL54B 49797127 IC50 = 3900 nM T50773 C5OUQ3 49797128 IC50 = 15000 nM T50773 C25ZSD 49797191 IC50 = 1400 nM T50773 C0OJX9 49797192 IC50 = 1400 nM T50773 C7GZ4B 49797193 IC50 = 160 nM T50773 CVT2E5 49797194 IC50 = 3500 nM T50773 C75MGE 49797195 IC50 = 1700 nM T50773 CVS70C 49797196 IC50 = 3700 nM T50773 C42QPW 49797197 IC50 = 44800 nM T50773 C6ZGL5 49797198 IC50 = 20400 nM T50773 C1B5NH 49797199 IC50 = 2920 nM T50773 CGQN24 49797200 IC50 = 850 nM T50773 CS2AI5 49797201 IC50 = 4200 nM T50773 CM7RE3 49797202 IC50 = 1050 nM T50773 CGM9E7 49797203 IC50 = 5410 nM T50773 COU0I6 49797204 IC50 = 2570 nM T50773 C3XML2 49797205 IC50 = 1700 nM T50773 CP0O2F 49797223 IC50 = 5500 nM T50773 CTH7I8 49797224 IC50 = 50000 nM T50773 CG9P7O 49797225 IC50 = 82000 nM T50773 C3A2QK 49797226 IC50 = 46000 nM T50773 C4NOK2 49797227 IC50 = 5300 nM T50773 CB13PO 49797228 IC50 = 28000 nM T50773 C47VOG 49797229 IC50 = 77000 nM T50773 CD2CL1 49797230 IC50 = 57000 nM T50773 C0LK6B 49797231 IC50 = 40000 nM T50773 CON0A6 49797232 IC50 > 100000 nM T50773 C4AVU3 49797233 IC50 = 54000 nM T50773 CQ93MI 49797234 IC50 = 33000 nM T50773 CO2JV8 49797235 IC50 > 100000 nM T50773 C27LDC 49797236 IC50 = 21000 nM T50773 CA5GM6 49797237 IC50 = 32000 nM T50773 CT8PW1 49797238 IC50 = 35000 nM T50773 CJQ38S 49797239 IC50 = 27000 nM T50773 CT65MR 49797240 IC50 = 58000 nM T50773 C08IFZ 49797241 IC50 = 87000 nM T50773 CA4E8M 49797242 IC50 = 93000 nM T50773 CN8FR2 49797243 IC50 = 64000 nM T50773 C37MDP 49797244 IC50 > 100000 nM T50773 CM41RN 49797245 IC50 = 41000 nM T50773 C59JEK 49797246 IC50 = 9900 nM T50773 CUMH43 49797248 IC50 > 100000 nM T50773 CM59PE 49797249 IC50 = 57000 nM T50773 CN5K1S 49797250 IC50 > 100000 nM T50773 CT5HY0 49797251 IC50 = 90000 nM T50773 C0E5PY 49797252 IC50 = 96000 nM T50773 C3E5JB 49797253 IC50 = 15000 nM T50773 CA8P5N 49797344 IC50 = 80000 nM T50773 CJL2B8 49797345 IC50 > 100000 nM T50773 CT79YI 49797346 IC50 > 100000 nM T50773 C93VJO 49797347 IC50 > 100000 nM T50773 CDI52A 49797348 IC50 = 4700 nM T50773 C7ATK9 49797349 IC50 > 100000 nM T50773 C2Y3DS 49797350 IC50 = 70000 nM T50773 CA4CE3 49797351 IC50 > 100000 nM T50773 C3A8YT 49797352 IC50 = 22000 nM T50773 C3HU6X 49797446 IC50 = 3440 nM T50773 C3U1KQ 49797450 IC50 = 1660 nM T50773 C76KMB 49797451 IC50 = 6400 nM T50773 C02MPV 49797452 IC50 = 15000 nM T50773 CLVF17 49797501 IC50 > 20000 nM T50773 CR0AK2 49797502 IC50 = 12000 nM T50773 CM1Y7K 49797503 IC50 > 20000 nM T50773 CUSI73 49797504 IC50 > 20000 nM T50773 CJ0DX6 49797505 IC50 > 20000 nM T50773 C2A7LE 49797506 IC50 > 20000 nM T50773 CU4M3T 49797507 IC50 > 20000 nM T50773 C8GCS5 49797508 IC50 > 20000 nM T50773 CTP9L2 49797509 IC50 > 20000 nM T50773 CT76PM 49797510 IC50 > 20000 nM T50773 C4K0QT 49797511 IC50 = 17000 nM T50773 CC56FE 49797513 IC50 > 20000 nM T50773 C4T6AB 49797514 IC50 > 20000 nM T50773 C41VHF 49797515 IC50 > 20000 nM T50773 CBD9H2 49797516 IC50 > 20000 nM T50773 CAOC90 49797517 IC50 > 20000 nM T50773 C0F5QX 49797518 IC50 > 20000 nM T50773 C7T5XW 49797519 IC50 > 20000 nM T50773 CM6SF5 49797520 IC50 > 20000 nM T50773 CQZN45 49797521 IC50 > 20000 nM T50773 CG64BU 49797522 IC50 > 20000 nM T50773 C5G3MA 49797524 IC50 = 10000 nM T50773 CO42DE 49797525 IC50 = 4500 nM T50773 C5L1EP 49797526 IC50 = 12000 nM T50773 CTWR80 49797527 IC50 = 12000 nM T50773 CPIC42 49797528 IC50 > 20000 nM T50773 C5N1ZB 49797529 IC50 = 4500 nM T50773 CU72EZ 49797596 IC50 = 23000 nM T50773 C6AZ2C 49797599 IC50 = 98000 nM T50773 CR86PO 49797604 IC50 = 6500 nM T50773 C6DJX7 49797605 IC50 = 88000 nM T50773 CK3ZI1 49797607 IC50 = 74000 nM T50773 C7AD0C 49797610 IC50 = 22000 nM T50773 C4XHO5 49797612 IC50 > 100000 nM T50773 C7VL5U 49797614 IC50 = 73000 nM T50773 CY09JE 49797615 IC50 = 8300 nM T50773 C1ZLF0 49797616 IC50 > 100000 nM T50773 CN48OE 49797627 IC50 = 16000 nM T50773 CV6I0O 49797630 IC50 = 41000 nM T50773 CAG1U7 49797631 IC50 > 100000 nM T50773 C8JNU1 49797636 IC50 = 22000 nM T50773 C0DN5G 49797642 IC50 = 2300 nM T50773 CJVS96 49797644 IC50 = 33000 nM T50773 CBRT78 49797650 IC50 = 54000 nM T50773 CZW93Y 49797653 IC50 = 5500 nM T50773 C85CEJ 51346970 IC50 = 63000 nM T50773 C4PFT3 51346971 IC50 = 8500 nM T50773 C7RJM9 52945660 IC50 = 2600 nM T50773 CC56BV 52946866 IC50 > 100000 nM T50773 CYC69Q 53317564 IC50 = 9600 nM T50773 C0QOV9 53317565 IC50 = 23000 nM T50773 CURC70 53317566 IC50 = 29000 nM T50773 C3ZK1W 53317575 IC50 = 83000 nM T50773 CBQ0J7 53317579 IC50 = 18000 nM T50773 CIY9F7 53317580 IC50 = 54000 nM T50773 C5DMS9 53317581 IC50 = 66000 nM T50773 C1XD9W 53317582 IC50 = 11000 nM T50773 CR0O8T 53317583 IC50 = 22000 nM T50773 C9GLH7 53318841 IC50 = 15000 nM T50773 C06TDE 53318842 IC50 = 17000 nM T50773 C73TER 53318856 IC50 = 35000 nM T50773 CC56NE 53318863 IC50 = 17000 nM T50773 C4UJI8 53318864 IC50 = 72000 nM T50773 C8CZ2A 53318865 IC50 = 52000 nM T50773 CLVY47 53318866 IC50 = 85000 nM T50773 CM7S5W 53319067 IC50 = 37000 nM T50773 C1X3NE 53320178 IC50 = 18000 nM T50773 C1P8BK 53320179 IC50 = 3600 nM T50773 C50UBZ 53320180 IC50 = 21000 nM T50773 C2JTR7 53320181 IC50 > 100000 nM T50773 C0TYJ5 53320182 IC50 = 39000 nM T50773 C7RSX2 53320183 IC50 = 48000 nM T50773 C9XGE4 53321472 IC50 = 19000 nM T50773 CY0ZV9 53321485 IC50 = 43000 nM T50773 CK0OB2 53321486 IC50 = 29000 nM T50773 CNK34J 53321487 IC50 = 68000 nM T50773 C7EO3D 53321495 IC50 = 32000 nM T50773 C3M7PQ 53321496 IC50 = 16000 nM T50773 C0NUQ7 53321497 IC50 = 17000 nM T50773 C31DSJ 53321498 IC50 = 19000 nM T50773 C2ZKV9 53321499 IC50 = 28000 nM T50773 CB76JK 53321550 IC50 > 30000 nM T50773 C3QT0R 53321621 IC50 = 20000 nM T50773 CXIS21 53322758 IC50 > 100000 nM T50773 CY71QL 53322814 IC50 > 100000 nM T50773 CLU96Y 53322820 IC50 > 100000 nM T50773 C8YVF1 53322821 IC50 = 12000 nM T50773 C4QS6V 53322822 IC50 = 14000 nM T50773 C62JTB 53322823 IC50 = 27000 nM T50773 CT14FU 53322824 IC50 = 23000 nM T50773 CXJ1F8 53322825 IC50 = 30000 nM T50773 C3K1VY 53322826 IC50 = 23000 nM T50773 C9N6HK 53322952 IC50 = 11000 nM T50773 C9LU8M 53324129 IC50 = 20000 nM T50773 CCY7M0 53324130 IC50 = 13000 nM T50773 C4F1QK 53324142 IC50 > 100000 nM T50773 CZN71C 53324143 IC50 = 10000 nM T50773 CG83JZ 53324144 IC50 > 100000 nM T50773 CE8J1D 53324145 IC50 = 58000 nM T50773 C0Y3AC 53324153 IC50 = 58000 nM T50773 C9O1IW 53324154 IC50 = 4800 nM T50773 CTW5G0 53324155 IC50 = 65000 nM T50773 C2DPZ0 53324156 IC50 = 13000 nM T50773 CL5Z8N 53324211 IC50 > 30000 nM T50773 CSN28M 53324293 IC50 = 86000 nM T50773 C25OJW 53325399 IC50 = 34000 nM T50773 CXW5O9 53325446 IC50 = 57000 nM T50773 C1SO0C 53325447 IC50 = 40000 nM T50773 C1S3WB 53325453 IC50 = 80000 nM T50773 C2KFW6 53325454 IC50 = 35000 nM T50773 C4ZFR5 53325455 IC50 = 42000 nM T50773 CV0H8P 53326691 IC50 = 20000 nM T50773 C3ZWN6 53326704 IC50 = 34000 nM T50773 C73SKG 53326705 IC50 = 11000 nM T50773 CG9V4W 53326706 IC50 = 81000 nM T50773 C5K8CP 53326713 IC50 = 51000 nM T50773 CN12AO 53353383 IC50 > 100000 nM T50773 C51GUC 53354365 IC50 > 100000 nM T50773 CRJ5P9 53354369 IC50 > 100000 nM T50773 C4G2HT 53354470 IC50 > 100000 nM T50773 C5P9VZ 53465973 IC50 = 19300 nM T50773 C7OBF2 53465974 IC50 = 14000 nM T50773 CF5YJ8 53465975 IC50 > 100000 nM T50773 C5XER7 53466046 IC50 > 25000 nM T50773 CJ9T8M 53466047 IC50 > 50000 nM T50773 CP1CL8 53466049 IC50 > 25000 nM T50773 CPSQ16 53466050 IC50 > 100000 nM T50773 C4UC1P 53466119 IC50 = 3300 nM T50773 C59SML 53466121 IC50 > 25000 nM T50773 C7JPY2 53466122 IC50 > 50000 nM T50773 CYZK63 53466123 IC50 > 25000 nM T50773 CVJ0D5 53466193 IC50 = 1900 nM T50773 C2XE8Y 53466195 IC50 > 25000 nM T50773 C0P2YE 53466196 IC50 > 25000 nM T50773 CPA0K4 53466271 IC50 > 100000 nM T50773 CYG36O 53466361 IC50 = 3600 nM T50773 C8U4OD 56649692 IC50 > 1000000 nM T50773 C1QX0O 56657809 IC50 > 100000 nM T50773 CU74VH 56658024 IC50 = 23000 nM T50773 CF6PV5 56658026 IC50 = 2100 nM T50773 C2KI8Y 56658028 IC50 = 170 nM T50773 CY4E6U 56658138 IC50 = 15200 nM T50773 C1PI4L 56664962 IC50 = 650 nM T50773 C8GPO1 56665883 IC50 = 730 nM T50773 CXH5W7 56671896 IC50 = 17300 nM T50773 CBK31U 56675279 IC50 = 33 nM T50773 CW8KU6 56675536 IC50 > 50000 nM T50773 C9ZE7J 58874273 IC50 > 10000 nM T50773 CW64RD 66561555 IC50 > 100000 nM T50773 C9GTI7 66561556 IC50 > 100000 nM T50773 C6HRX1 68845950 IC50 = 6600 nM T50773 C5W6LY 70681316 IC50 > 100000 nM T50773 CLO96S 70681357 IC50 > 100000 nM T50773 CWP41T 70681469 IC50 > 100000 nM T50773 C7Z2KY 70681470 IC50 > 100000 nM T50773 C19XIQ 70683454 IC50 > 100000 nM T50773 C07ADL 70683455 IC50 > 100000 nM T50773 CO2NK6 70685557 IC50 > 100000 nM T50773 CK0WX8 70685558 IC50 > 100000 nM T50773 CLF84U 70685559 IC50 > 100000 nM T50773 C0K7PS 70685560 IC50 > 100000 nM T50773 C2T0NS 70685696 IC50 > 100000 nM T50773 CVD76F 70687705 IC50 > 100000 nM T50773 C28GVW 70687706 IC50 > 100000 nM T50773 CVYH31 70689717 IC50 > 100000 nM T50773 CUY81P 70689750 IC50 > 100000 nM T50773 CX2O0Z 70689751 IC50 > 100000 nM T50773 C17YKW 70689752 IC50 = 23300 nM T50773 C87LMG 70691901 IC50 > 100000 nM T50773 CL5EG7 70691902 IC50 > 100000 nM T50773 CGND49 70691903 IC50 > 100000 nM T50773 CGT57B 70691904 IC50 > 100000 nM T50773 CT89CW 70691905 IC50 > 100000 nM T50773 C5WI6V 70691906 IC50 > 100000 nM T50773 CQMV53 70693949 IC50 > 100000 nM T50773 CBP8U7 70693950 IC50 > 100000 nM T50773 C0I2CV 70693951 IC50 > 100000 nM T50773 CCB64G 70693952 IC50 > 100000 nM T50773 C3ZUK2 70693953 IC50 > 100000 nM T50773 CS76EN 70693954 IC50 > 100000 nM T50773 C27PFC 70693955 IC50 > 100000 nM T50773 CVY48R 70693956 IC50 > 100000 nM T50773 CA01KO 70696068 IC50 > 100000 nM T50773 CSW43K 70696069 IC50 > 100000 nM T50773 C19ZWC 70789754 IC50 > 100000 nM T50773 CP91OE 71203742 IC50 > 100000 nM T50773 CP6G5W 71203746 IC50 > 100000 nM T50773 C32UMV 71203748 IC50 > 100000 nM T50773 C04XQY 71203752 IC50 > 100000 nM T50773 CE2I0K 71203758 IC50 > 100000 nM T50773 C5GEJ9 71203769 IC50 > 100000 nM T50773 C7LKV0 71203783 IC50 > 100000 nM T50773 CM5DB6 71450086 IC50 > 100000 nM T50773 CQU0Z1 71450087 IC50 > 100000 nM T50773 C65BCE 71450089 IC50 > 10000 nM T50773 CP9K2W 71450603 IC50 = 4600 nM T50773 CLC2N8 71451900 IC50 > 100000 nM T50773 CMU63C 71451901 IC50 > 100000 nM T50773 CT5WU4 71451902 IC50 > 100000 nM T50773 CL0X3F 71451939 IC50 > 100000 nM T50773 C61LNR 71452448 IC50 = 6700 nM T50773 CEM2O9 71453723 IC50 > 100000 nM T50773 CB1EX7 71453762 IC50 > 100000 nM T50773 CN4FE7 71454208 IC50 = 8600 nM T50773 CBOK64 71455456 IC50 > 100000 nM T50773 CD32GT 71455458 IC50 > 100000 nM T50773 CQA9L7 71455494 IC50 > 100000 nM T50773 C1LRH5 71455960 IC50 = 34600 nM T50773 C4T7CO 71457236 IC50 > 100000 nM T50773 C3GAO1 71457237 IC50 > 100000 nM T50773 CE3MP2 71457238 IC50 > 100000 nM T50773 C42BSO 71457239 IC50 > 100000 nM T50773 C8VI9L 71457240 IC50 > 100000 nM T50773 C59TGZ 71457761 IC50 = 2700 nM T50773 C5T6QP 71457765 IC50 = 45400 nM T50773 CIO50T 71459090 IC50 > 10000 nM T50773 CXIM97 71459091 IC50 > 100000 nM T50773 CJ6N1C 71459092 IC50 > 100000 nM T50773 CUB4V8 71459679 IC50 = 1700 nM T50773 CSC3I7 71460901 IC50 > 100000 nM T50773 CG7VX2 71460902 IC50 > 10000 nM T50773 C5K3WJ 71460903 IC50 > 100000 nM T50773 C3UF9P 71460904 IC50 > 100000 nM T50773 C7TS9F 71462596 IC50 > 100000 nM T50773 C63SUR 71462597 IC50 > 100000 nM T50773 CZT3S0 71462641 IC50 > 100000 nM T50773 CKZ17B 71463121 IC50 = 22000 nM T50773 C4VKM3 71463122 IC50 = 29400 nM T50773 C7B8AO 71621488 IC50 > 100000 nM T50773 CC93KJ 71655554 IC50 > 100000 nM T50773 CN90KH 71655555 IC50 > 100000 nM T50773 CUT37D 71655556 IC50 > 100000 nM T50773 C71OFQ 71655557 IC50 > 100000 nM T50773 C7R6HU 71655622 IC50 > 100000 nM T50773 C2NA1M 71655623 IC50 > 100000 nM T50773 CDF08H 71655624 IC50 > 100000 nM T50773 CBEX27 71655625 IC50 > 100000 nM T50773 CT6XB5 71655626 IC50 > 100000 nM T50773 C1ND2P 71655627 IC50 > 100000 nM T50773 CXZ8N4 71667081 IC50 > 100000 nM T50773 CJ9QU7 71667226 IC50 > 100000 nM T50773 CE0Z8G 71667227 IC50 > 100000 nM T50773 CL7CS3 71667230 IC50 > 100000 nM T50773 CB6SI5 71667231 IC50 > 100000 nM T50773 C75UWV 71667375 IC50 > 100000 nM T50773 C19CTI 71667376 IC50 > 100000 nM T50773 C69CJB 71667378 IC50 > 100000 nM T50773 C07HNK 71667379 IC50 > 100000 nM T50773 CK74SP 71667380 IC50 > 100000 nM T50773 CMYZ68 71667381 IC50 > 100000 nM T50773 CDI39U 71667510 IC50 > 100000 nM T50773 C7BD2R 71720854 IC50 = 8400 nM T50773 C9Q8MO 72164809 IC50 = 640 nM T50773 CL5X1Z 72164811 IC50 = 1030 nM T50773 C7N8WB 72164813 IC50 = 1880 nM T50773 C2R0NV 72164815 IC50 = 340 nM T50773 C4JLM5 72164817 IC50 = 440 nM T50773 C6RQ9A 72164819 IC50 = 1040 nM T50773 C38GWP 72164942 IC50 = 930 nM T50773 C4T0MY 72164944 IC50 = 520 nM T50773 C0T4UW 72164946 IC50 = 1460 nM T50773 CLV02R 72164948 IC50 = 1200 nM T50773 CHPN10 72164950 IC50 = 2520 nM T50773 CI78FQ 72165082 IC50 = 1100 nM T50773 CN0VU2 72165084 IC50 = 2090 nM T50773 C84SYX 72165086 IC50 = 660 nM T50773 C1RQA3 72165088 IC50 = 570 nM T50773 CH51ZR 72165090 IC50 = 1560 nM T50773 C1HL2A 72188903 IC50 = 15400 nM T50773 CLS1A0 72188904 IC50 > 100000 nM T50773 CO15AV 72188905 IC50 = 19000 nM T50773 CPDC28 72188906 IC50 = 160 nM T50773 CL7P3D 72193502 IC50 > 100000 nM T50773 C4AXB8 72193503 IC50 > 100000 nM T50773 CQC28P 72193504 IC50 > 100000 nM T50773 CV87PE 72193505 IC50 > 100000 nM T50773 C65DFP 72697059 IC50 = 296900 nM T50773 CX07OC 72697060 IC50 = 5440 nM T50773 CZ56DO 72697061 IC50 = 5880 nM T50773 C1A2KX 72697062 IC50 = 8780 nM T50773 CS5U1F 72697063 IC50 = 4670 nM T50773 CA3HI1 72697064 IC50 = 1700 nM T50773 CCZJ47 72697206 IC50 = 2140 nM T50773 CWNZ91 72697207 IC50 = 1570 nM T50773 C6BWI4 72697208 IC50 = 7010 nM T50773 C9JA1Q 72697209 IC50 = 6220 nM T50773 CF6A8N 72697210 IC50 = 4110 nM T50773 CC7G3M 72697353 IC50 = 1320 nM T50773 CXYO73 72697354 IC50 = 1700 nM T50773 CAXV78 72697355 IC50 = 14520 nM T50773 CGV09W 72697356 IC50 = 1440 nM T50773 CIF9D7 72697357 IC50 = 1720 nM T50773 CC8RA6 72697358 IC50 = 1440 nM T50773 C1EC7S 72697359 IC50 = 39090 nM T50773 C8CRO6 72697494 IC50 = 800 nM T50773 CP0MU3 72697496 IC50 = 1080 nM T50773 CI60AK 72697497 IC50 = 120 nM T50773 CO19YK 72697498 IC50 = 100000 nM T50773 C47IGZ 72697499 IC50 = 102000 nM T50773 C65OPG 72697500 IC50 = 1810 nM T50773 C3ZP7N 72697501 IC50 = 2540 nM T50773 C7EF8C 72697646 IC50 = 1290 nM T50773 CC10AZ 73345857 IC50 > 100000 nM T50773 CSZR98 73346173 IC50 = 11000 nM T50773 C1L4RX 73346174 IC50 = 38000 nM T50773 CX4F0Y 73347359 IC50 > 100000 nM T50773 C3XFM5 73347360 IC50 > 100000 nM T50773 CGNL10 73347698 IC50 > 100000 nM T50773 CR09PJ 73348871 IC50 > 10000 nM T50773 CO5TB8 73349220 IC50 > 100000 nM T50773 C06WRM 73350448 IC50 > 100000 nM T50773 C1T7LK 73350449 IC50 > 100000 nM T50773 CCIZ12 73350450 IC50 > 100000 nM T50773 CNC6B8 73350798 IC50 = 65000 nM T50773 CDBV29 73350799 IC50 = 70000 nM T50773 CYG04J 73352283 IC50 = 3900 nM T50773 CFV5U3 73353424 IC50 > 100000 nM T50773 CRS4O0 73353425 IC50 > 100000 nM T50773 CV6BA3 73353756 IC50 > 100000 nM T50773 C51QGP 73353757 IC50 = 15000 nM T50773 CBK37N 73353758 IC50 > 100000 nM T50773 CLYP23 73354936 IC50 > 100000 nM T50773 CLO76J 73355285 IC50 > 100000 nM T50773 CCVT96 73355286 IC50 > 100000 nM T50773 CH9W2R 73356494 IC50 > 100000 nM T50773 CKD46T 73356495 IC50 > 100000 nM T50773 CI0N6E 73356496 IC50 > 10000 nM T50773 CB60OP 89488720 IC50 > 100000 nM T50773 CIV7Y8 89668929 IC50 > 100000 nM T50773 C87GJT 89704940 IC50 > 100000 nM T50773 CHI7U9 89704942 IC50 > 100000 nM T50773 CSLI09 89704955 IC50 > 100000 nM T50773 CA3K7R 89704970 IC50 > 100000 nM T50773 CF89OD 89705045 IC50 > 100000 nM T50773 CK3Z8J 89705076 IC50 > 100000 nM T50773 CH6P0S 89705081 IC50 > 100000 nM T50773 C63DGS 89705096 IC50 > 100000 nM T50773 CND56S 89705098 IC50 > 100000 nM T50773 C0CKQ7 89705100 IC50 > 100000 nM T50773 C0CPD1 89705103 IC50 > 100000 nM T50773 C1IL7N 89705109 IC50 > 100000 nM T50773 CA48MR 89705136 IC50 > 100000 nM T50773 C5F9OA 89705152 IC50 > 50000 nM T50773 C1VSG5 89705179 IC50 > 100000 nM T50773 CHAS49 89705195 IC50 > 100000 nM T50773 C0RP1J 89705223 IC50 > 100000 nM T50773 CQO0I6 89705242 IC50 > 100000 nM T50773 C7DF1P 89705244 IC50 > 100000 nM T50773 C03OGJ 89705273 IC50 > 100000 nM T50773 CGX4I7 89705275 IC50 > 100000 nM T50773 CX9BC3 89712515 IC50 > 100000 nM T50773 C6TGZ5 90655538 IC50 > 100000 nM T50773 C9P3HJ 90655539 IC50 > 100000 nM T50773 CT98OM 90655540 IC50 > 100000 nM T50773 CVQ8M4 90655541 IC50 > 100000 nM T50773 CT6Q2L 90655542 IC50 > 100000 nM T50773 C7Z4GV 90655543 IC50 > 100000 nM T50773 CE3HC2 90655544 IC50 > 100000 nM T50773 CU2I3V 90655545 IC50 > 100000 nM T50773 C2NZ7X 90655546 IC50 > 100000 nM T50773 C0E5UP 90655547 IC50 > 100000 nM T50773 CF23RI 90655548 IC50 > 100000 nM T50773 CW3QG7 90655549 IC50 > 100000 nM T50773 CHG4E2 90655550 IC50 > 100000 nM T50773 CTA78W 90655551 IC50 > 100000 nM T50773 CA6S4W 90655552 IC50 > 100000 nM T50773 C3LT0S 90655553 IC50 > 100000 nM T50773 CEW45X 90655554 IC50 > 100000 nM T50773 CRX52D 90655555 IC50 > 100000 nM T50773 C9KG1U 90655556 IC50 > 100000 nM T50773 CXYE76 90655557 IC50 > 100000 nM T50773 CES85Q 90655558 IC50 > 100000 nM T50773 CK7IB9 90655559 IC50 > 100000 nM T50773 CAG5X4 90655560 IC50 > 100000 nM T50773 C3IJA0 90655561 IC50 > 100000 nM T50773 C4V0ZY 90655562 IC50 > 100000 nM T50773 CY9G8Q 90655563 IC50 > 50000 nM T50773 CU9LB2 90664438 IC50 > 25000 nM T50773 CQ20XA 90664578 IC50 = 290 nM T50773 CV87ZH 90664579 IC50 > 50000 nM T50773 CDEN13 90664693 IC50 > 50000 nM T50773 CV0SF5 90664925 IC50 > 10000 nM T50773 CBQ38C 101879512 IC50 = 207350 nM T50773 CM7E4V 101887269 IC50 > 100000 nM T50773 C8EH0J 101887270 IC50 > 100000 nM T50773 CDT67J 101887271 IC50 > 100000 nM T50773 C4F2CS 101887272 IC50 > 100000 nM T50773 C58XWA 101887273 IC50 > 100000 nM T50773 C3Y9ET 101887274 IC50 > 100000 nM T50773 C1AF8C 101887275 IC50 > 100000 nM T50773 CH7QC5 101887276 IC50 > 100000 nM T50773 CO4FR2 101887277 IC50 > 100000 nM T50773 C9JEH0 101887278 IC50 > 100000 nM T50773 C52GIO 101887279 IC50 > 100000 nM T50773 C3W5RU 118712765 IC50 = 129710 nM T50773 C8M6ZW 118712767 IC50 = 59100 nM T50773 CV5C6D 118712768 IC50 = 192790 nM T50773 C2NSC7 118712769 IC50 = 9550 nM T50773 CAR4W5 118712772 IC50 = 31800 nM T50773 CRWT85 118712773 IC50 = 9340 nM T50773 C4T2FY 118712775 IC50 = 50620 nM T50773 CD0HQ4 118712781 IC50 = 77030 nM T50773 C46TMQ 118712785 IC50 = 28260 nM T50773 C5M3BX 118712788 IC50 = 71680 nM T50773 CK71WT 118722410 IC50 = 31940 nM T50773 CI74ZM 118722411 IC50 = 23100 nM T50773 CH1P7Y 118722412 IC50 = 24340 nM T50773 C8KUP0 118722416 IC50 = 6850 nM T50773 COG4V6 118722421 IC50 = 14000 nM T50773 CN78TQ 122189864 IC50 > 100000 nM T50773 CNM82F 122189865 IC50 > 100000 nM T50773 C19GHJ 122189866 IC50 > 100000 nM T50773 C3U9KC 122189867 IC50 > 100000 nM T50773 CW5V3U 122189868 IC50 > 100000 nM T50773 CCG05R 122189869 IC50 > 100000 nM T50773 CI01PT 122189870 IC50 > 100000 nM T50773 C80EWF 122189871 IC50 > 100000 nM T50773 C3N7JC 122189872 IC50 > 100000 nM T50773 CG8O1J 122189873 IC50 > 100000 nM T50773 CK0US2 122189874 IC50 > 100000 nM T50773 C5V6NI 122189875 IC50 > 100000 nM T50773 CV7A9Y 122189876 IC50 > 100000 nM T50773 CH97SN 122189877 IC50 > 100000 nM T50773 CN86VR 122189878 IC50 > 100000 nM T50773 CZB49I 122189879 IC50 > 100000 nM T50773 C6PLX9 127035081 IC50 = 33000 nM T50773 CJ0KS7 127035239 IC50 > 100000 nM T50773 CKSZ13 127035240 IC50 > 100000 nM T50773 C6T1IM 127035241 IC50 > 100000 nM T50773 CJRL72 127035242 IC50 > 100000 nM T50773 CVKI59 127035243 IC50 = 61000 nM T50773 CWJX95 127035244 IC50 = 95000 nM T50773 C0XMS7 127035375 IC50 > 100000 nM T50773 CMK5Q9 127035376 IC50 > 100000 nM T50773 C4N7QB 127035377 IC50 > 100000 nM T50773 CGN49F 127035378 IC50 = 70000 nM T50773 C36UHW 127035569 IC50 = 44000 nM T50773 CTKS36 127035740 IC50 > 100000 nM T50773 CAXT02 127035741 IC50 > 100000 nM T50773 CZB0L6 127035742 IC50 = 57000 nM T50773 C4QWL5 127035743 IC50 > 100000 nM T50773 CPGF39 127035744 IC50 > 100000 nM T50773 CXTD34 127035745 IC50 = 88000 nM T50773 CM98XR 127035752 IC50 > 100000 nM T50773 C87MVA 127035753 IC50 > 100000 nM T50773 CDW25O 127035754 IC50 = 27000 nM T50773 CN08IS 127045827 IC50 > 100000 nM T50773 CAK85G 127046590 IC50 > 100000 nM T50773 CP3U8J 127046622 IC50 = 31000 nM T50773 CFAI71 127046624 IC50 = 9400 nM T50773 CB6PA7 127046626 IC50 > 100000 nM T50773 C76IGF 127046628 IC50 > 100000 nM T50773 CHL49F 127046630 IC50 = 22000 nM T50773 CH0D2Z 127046632 IC50 > 100000 nM T50773 CK4SO7 127047730 IC50 = 1100 nM T50773 CSO9L3 127047731 IC50 = 23000 nM T50773 C4KIA9 127047732 IC50 = 12900 nM T50773 CHX41E 127047733 IC50 = 25 nM T50773 C6I7HW 127047734 IC50 > 100000 nM T50773 C2CP4F 127047761 IC50 = 40000 nM T50773 CYR1X2 127047762 IC50 > 100000 nM T50773 CIV4C2 127047839 IC50 > 25000 nM T50773 CDYA70 127047985 IC50 = 14800 nM T50773 C0FS5E 127048116 IC50 = 10900 nM T50773 CRM4Q8 135518358 IC50 = 1100 nM T50773 CMI5A6 135964368 IC50 = 1100 nM T50773 CO04QA 136177302 IC50 = 46000 nM T50773 D02RDY 11375559 IC50 = 38377 nM T50773 D03DNV 71655266 IC50 > 100000 nM T50773 D07ALM 11232124 Ki = 0.082 nM T50773 D07IJU 13578534 IC50 > 500000 nM T50773 D0CP1J 56658139 IC50 > 1000000 nM T50773 D0L5RI 44328273 Ki = 277 nM T50773 D0L9XR 447256 IC50 = 153000 nM T50773 D0N1FU 6918465 Ki = 8170 nM T50773 D0T2EW 11075394 IC50 = 39873 nM T29683 D0GU4K 135413536 Ki = 454.1 nM T29683 D02IWC 23649245 IC50 = 1.6 nM T29683 D05ZWG 108147 EC50 = 0.0034 nM T29683 D0CB2B 23653789 Ki = 2.4 nM T29683 D0K5HI 5311424 Ki = 1 nM T29683 D00VPT 6604009 Ki = 3.8 nM T29683 D02TKI 132846 IC50 > 1000 nM T29683 D03SXN 104943 Ki > 10000 nM T29683 D08ZBV 132837 IC50 > 5000 nM T29683 D0IP6X 219077 Ki = 0.1995 nM T29683 D0J3QU 44351946 Ki = 9190 nM T29683 D0N1PA 9869033 IC50 = 2650 nM T29683 CIG4C3 132957 EC50 = 10.88 nM T29683 CC8X2D 133090 Ki = 2.4 nM T29683 C20AYU 153996 Ki = 200 nM T29683 C4NS9E 667698 Ki = 355 nM T29683 C5N1KX 1760285 Ki = 18 nM T29683 CMLC05 1760287 Ki = 13.8 nM T29683 C9T8LQ 1981061 Ki = 134 nM T29683 CBR7A4 2314026 Ki = 6208 nM T29683 CQEC49 2932589 Ki = 31.62 nM T29683 CNX2V8 3245625 IC50 = 1100 nM T29683 C50GNY 3628880 Ki = 3162.28 nM T29683 CQW7N2 3946663 Ki = 10 nM T29683 C0UR7K 4529080 Ki = 30.7 nM T29683 C5PO1F 6604014 Ki = 13.3 nM T29683 CE57YD 6604858 Ki = 13 nM T29683 C36VYU 7016092 IC50 > 5000 nM T29683 CO5I6D 7033529 IC50 = 1500 nM T29683 C2W6PI 8867347 IC50 = 480 nM T29683 CMI05O 8870164 IC50 = 2100 nM T29683 CPRQ41 9806459 Ki = 193 nM T29683 CL81MT 9809876 Ki = 220 nM T29683 CIGT19 9810434 Ki = 0.5 nM T29683 C35MSJ 9810544 Ki = 0.3 nM T29683 CP38OJ 9825316 Ki = 3.4 nM T29683 C5Q8EM 9828448 Ki = 454 nM T29683 C07FWV 9830361 Ki = 1.7 nM T29683 CN6WE9 9831075 Ki = 0.7 nM T29683 C9BDV3 9831546 Ki = 0.4 nM T29683 CHIS10 9831674 Ki = 1.3 nM T29683 C3TV1U 9831707 Ki = 0.5 nM T29683 CZ46YW 9843873 Ki = 7.943 nM T29683 C52PUJ 9849950 Ki = 1210 nM T29683 CWEH02 9851237 IC50 = 39 nM T29683 CIXG30 9852376 IC50 = 25 nM T29683 CMZ20K 9852630 Ki = 0.8 nM T29683 C2JS5O 9852904 Ki = 9.4 nM T29683 CSU2Y3 9853636 Ki = 0.4 nM T29683 CY37UT 9853827 Ki = 1258.93 nM T29683 C3LOJ7 9872857 Ki = 1.9 nM T29683 CCE74U 9874473 Ki = 97 nM T29683 CD6U7Z 9875034 Ki = 0.3 nM T29683 CA2X8G 9875056 Ki = 0.5 nM T29683 CW07IY 9896757 Ki = 0.8 nM T29683 C4SEJ2 9917970 Ki = 0.6 nM T29683 CPZ4B5 9956370 Ki = 1250 nM T29683 CQ69EA 9957749 Ki > 12000 nM T29683 C7ZXS9 9958115 Ki = 1254 nM T29683 C0DZ6K 9961315 Ki = 39 nM T29683 CNP82Y 9961936 Ki = 2 nM T29683 C8CY0E 9961955 Ki = 0.5 nM T29683 CG67TC 9970049 Ki = 47.2 nM T29683 C7BG9Z 9981979 IC50 > 5000 nM T29683 CHA2I0 10000989 Ki = 3.981 nM T29683 C6SPN0 10001673 IC50 = 5200 nM T29683 C5ZY7C 10016461 IC50 = 9400 nM T29683 C1XK9Y 10019102 IC50 > 10000 nM T29683 C5LQ0J 10024953 IC50 = 60000 nM T29683 CH6DS8 10025594 IC50 > 5000 nM T29683 C10WEQ 10041813 IC50 > 5000 nM T29683 CGS3X5 10041814 IC50 > 5000 nM T29683 CEIQ93 10043484 IC50 > 5000 nM T29683 CVJ8O1 10045010 IC50 > 5000 nM T29683 C25WVJ 10047566 IC50 > 1000 nM T29683 CRN1L3 10047989 IC50 > 5000 nM T29683 C7KUO1 10071124 IC50 > 5000 nM T29683 CH5YG4 10072464 IC50 = 3000 nM T29683 C1WVZ0 10102903 EC50 = 0.013 nM T29683 CU6P3B 10113552 Ki = 2581 nM T29683 CB5T4E 10114860 Ki = 50.12 nM T29683 CA8Z7P 10135793 Ki = 924 nM T29683 C4QC6M 10136512 Ki = 96 nM T29683 C85XEY 10151946 Ki = 1999 nM T29683 CP6I0S 10155886 Ki = 199.53 nM T29683 CS68EB 10160182 Ki = 377 nM T29683 CU81IJ 10173872 Ki = 631 nM T29683 C1XB9M 10177878 Ki = 1.995 nM T29683 C4IU8G 10177949 Ki = 919 nM T29683 CW0BV3 10179239 Ki = 66 nM T29683 CFCI14 10179473 Ki = 454 nM T29683 CZCX69 10194796 Ki = 3815 nM T29683 CF07PG 10202481 Ki = 15.2 nM T29683 CSA32M 10216430 Ki = 4051 nM T29683 C4FP3M 10222132 Ki = 129 nM T29683 CNOR67 10222384 Ki = 5.8 nM T29683 C1S5IR 10223181 Ki = 12.59 nM T29683 C6NA8J 10225028 Ki = 4874 nM T29683 CRF91O 10249483 Ki = 49 nM T29683 CVQ23E 10258592 IC50 = 1.2 nM T29683 C4F7IQ 10270385 Ki = 870 nM T29683 CK6Q8U 10271147 Ki = 74.3 nM T29683 CLIC45 10272462 Ki = 132 nM T29683 CEC41V 10291688 Ki = 1671 nM T29683 C1TSQ7 10296362 Ki = 629 nM T29683 C9HR5S 10303099 Ki = 11.36 nM T29683 CB8S4N 10318477 IC50 > 5000 nM T29683 CWFB30 10323427 IC50 > 1000 nM T29683 CI5U8S 10336036 IC50 = 3500 nM T29683 C95XTE 10340761 IC50 = 16 nM T29683 COJ4A7 10342797 IC50 > 5000 nM T29683 CWO60K 10350626 EC50 = 0.063 nM T29683 CN8PA7 10357986 IC50 > 10000 nM T29683 CZ1J0B 10362340 IC50 > 5000 nM T29683 C92BEU 10364942 IC50 > 5000 nM T29683 C6BQR5 10369844 IC50 > 5000 nM T29683 CVQ03A 10370066 Ki = 0.8 nM T29683 CYSX27 10389807 IC50 > 5000 nM T29683 CXG7P5 10393390 IC50 = 1.5 nM T29683 C4KZW9 10404051 IC50 > 5000 nM T29683 C5EKJ8 10405990 IC50 = 8000 nM T29683 C49JLI 10410206 IC50 > 5000 nM T29683 CDNR80 10410322 IC50 > 5000 nM T29683 C7EYZ4 10412224 IC50 > 5000 nM T29683 CNX23Q 10429546 IC50 > 5000 nM T29683 CRX37K 10430798 Ki = 1202 nM T29683 C9JPG8 10435750 IC50 > 5000 nM T29683 CQ76AR 10460302 IC50 = 1690 nM T29683 CS57CU 10474902 IC50 > 5000 nM T29683 C31BTI 10477667 IC50 > 5000 nM T29683 CY07LB 10477952 IC50 > 5000 nM T29683 CTFZ13 10477953 IC50 > 5000 nM T29683 CO49AP 10478708 IC50 = 3000 nM T29683 CR8X3F 10486632 EC50 = 10.73 nM T29683 CUEJ53 10501724 Ki = 1235 nM T29683 C1P6MW 10504093 IC50 = 74 nM T29683 C0Q9KT 10522097 Ki = 6203 nM T29683 C7KEV6 10524687 Ki = 6.31 nM T29683 C2DCQ6 10526297 Ki = 15.9 nM T29683 C6LK4N 10530762 IC50 = 92 nM T29683 C2EWU0 10548730 Ki = 426 nM T29683 CYHO36 10550310 IC50 > 10000 nM T29683 CD0G5V 10552329 Ki = 31.2 nM T29683 CQU3Y9 10555683 IC50 = 28 nM T29683 CL9C6S 10571967 Ki = 314 nM T29683 C5OTZ7 10572714 Ki = 146 nM T29683 CGI1M0 10575877 IC50 > 10000 nM T29683 CSY15N 10577242 IC50 = 1200 nM T29683 C17XAV 10578353 IC50 = 4310 nM T29683 C71VDU 10595071 Ki = 295 nM T29683 CXT80F 10596000 Ki = 983 nM T29683 C9A2IO 10596077 Ki > 33000 nM T29683 CC94FT 10597773 Ki = 1926 nM T29683 CT7C0R 10598474 IC50 > 10000 nM T29683 CIY19L 10600223 Ki = 4.7 nM T29683 CKVM50 10600296 Ki = 10.7 nM T29683 C1R9LK 10602517 IC50 = 111 nM T29683 C8UEI1 10619783 Ki = 5.5 nM T29683 C47DMY 10621487 Ki = 488 nM T29683 CBX09E 10622303 IC50 > 10000 nM T29683 C2N4PK 10622339 Ki = 666 nM T29683 CMWH10 10623566 Ki = 5.7 nM T29683 C0J8HK 10640904 Ki = 10312 nM T29683 CZ14UN 10641303 Ki > 10000 nM T29683 CPC13R 10645347 Ki = 5181 nM T29683 C7AM3X 10646059 IC50 = 1830 nM T29683 C5WL0T 10649927 IC50 = 425 nM T29683 C1KAO8 10650335 IC50 = 439 nM T29683 CWG05K 10650463 IC50 = 162 nM T29683 CLOF45 10668461 Ki = 1.8 nM T29683 CZ1K3M 10691318 Ki = 1.4 nM T29683 CQU7N3 10693681 IC50 > 10000 nM T29683 C6YDF1 10693682 IC50 > 10000 nM T29683 C92CQP 10693708 Ki = 1853 nM T29683 CNRK24 10695575 Ki = 8.6 nM T29683 C3JWM0 10696939 Ki = 1.8 nM T29683 CQ7V4Z 10698860 IC50 = 119 nM T29683 CTXL54 10709778 Ki > 33000 nM T29683 C3LQ1X 10714925 Ki = 382 nM T29683 CJM5W4 10715765 Ki > 10000 nM T29683 C6F1TM 10716102 Ki = 180 nM T29683 CBPH04 10716491 Ki = 1154 nM T29683 C06UEJ 10717542 Ki = 820 nM T29683 C6TEF1 10717843 Ki = 3.3 nM T29683 CY9FS1 10718673 Ki = 4.6 nM T29683 C63HTU 10722506 IC50 = 31 nM T29683 C7R6JW 10739572 Ki = 2226 nM T29683 CCF41R 10740312 Ki = 142 nM T29683 C2N8MY 10743411 IC50 = 350 nM T29683 CV96SZ 10743412 IC50 = 52 nM T29683 C8OG9Q 10744303 IC50 = 43 nM T29683 C1OBF3 10744541 Ki = 1.2 nM T29683 C45ACY 10745164 IC50 = 1400 nM T29683 C4G9VT 10762413 Ki = 1.995 nM T29683 CZ3D9W 10763631 Ki = 26 nM T29683 CZ4L0I 10764865 Ki = 4.7 nM T29683 CJ9A7P 10764902 Ki = 786 nM T29683 C3EZ5D 10769339 IC50 = 106 nM T29683 C3M1QK 10786254 Ki = 8133 nM T29683 CFIE37 10786383 Ki = 77 nM T29683 CK5RH3 10788357 Ki = 234 nM T29683 C8ZRV6 10788556 Ki = 57 nM T29683 C6MQB1 10790452 Ki = 2 nM T29683 C7DVG0 10792233 Ki = 1.4 nM T29683 CD3XW5 10810808 Ki = 883 nM T29683 C5XWZ8 10812218 Ki = 2.2 nM T29683 CRV5N0 10812309 IC50 > 10000 nM T29683 CWI34S 10813099 Ki = 45.3 nM T29683 C35ANM 10833965 Ki = 118 nM T29683 CJ46PG 10835383 Ki = 973 nM T29683 CE08LU 10836148 IC50 = 1520 nM T29683 C0JLK6 10836149 IC50 > 10000 nM T29683 C9FEW7 10836803 Ki = 6.3 nM T29683 C93WDV 10837046 Ki = 37.2 nM T29683 COH20K 10837820 Ki = 7 nM T29683 CH53JC 10840329 Ki = 1.2 nM T29683 C4SBO9 10915140 IC50 > 10000 nM T29683 CAB10S 11239751 Ki = 7943.28 nM T29683 C2TC9K 11273015 Ki = 5.9 nM T29683 CZ90JO 11296094 Ki = 2.91 nM T29683 CN9B1I 11353915 Ki = 5.4 nM T29683 C85LYP 11430418 IC50 > 1000 nM T29683 C8Z9SV 11467400 Ki = 12.22 nM T29683 C5USE7 11490769 Ki = 0.7 nM T29683 CY8T6X 11498183 Ki = 6.1 nM T29683 C0CUH7 11517160 IC50 = 210 nM T29683 C56TVA 11526802 Ki = 36 nM T29683 C7B0FA 11569867 Ki = 1 nM T29683 C6I1ML 11597466 IC50 = 7.4 nM T29683 COI0G2 11605470 IC50 = 11 nM T29683 CZH2M1 11618471 IC50 = 10 nM T29683 C5DPH7 11633686 IC50 = 53 nM T29683 C9X6JV 11657014 Ki = 83 nM T29683 CVM6L9 11676652 IC50 = 33 nM T29683 C7SE1K 11685645 Ki = 4.2 nM T29683 CA98DC 11794168 Ki = 25.12 nM T29683 CGBH98 11795836 Ki = 1078 nM T29683 C7QIR6 11797202 Ki = 180 nM T29683 CO19LD 11798897 Ki = 6.8 nM T29683 CV2FP5 11800009 IC50 = 1080 nM T29683 CX7S5D 11800732 Ki = 1.5 nM T29683 C2Q1AP 11818775 EC50 = 0.079 nM T29683 CZ9FS3 11990142 IC50 = 7.4 nM T29683 C0OU2J 15485361 IC50 = 19 nM T29683 COJ24C 15508105 Ki = 10 nM T29683 CI5O7S 15608404 IC50 = 28 nM T29683 CWH6F8 16035466 IC50 = 5.2 nM T29683 CY8LG6 16036824 EC50 = 36 nM T29683 C3P9FH 16064397 EC50 = 2.5 nM T29683 CWK98Z 16065257 EC50 = 4.9 nM T29683 CNYF14 16065390 EC50 = 14 nM T29683 C59BZD 16065391 EC50 = 6.9 nM T29683 CXGM03 16065392 EC50 = 35 nM T29683 CJ37FY 19572770 IC50 = 3810 nM T29683 C69KET 20864936 IC50 = 390 nM T29683 CA63LJ 20906556 IC50 = 240 nM T29683 C81JWV 20906619 IC50 = 130 nM T29683 CMEF68 20906620 IC50 > 10000 nM T29683 C8H7FU 20910781 IC50 > 10000 nM T29683 CXF8Z9 23294208 IC50 = 539 nM T29683 C3XN1D 23294214 IC50 = 7.9 nM T29683 CZ7V4E 24851680 Ki = 0.3981 nM T29683 CO9I3A 25181433 Ki = 10 nM T29683 CT5K8R 25195470 Ki = 0.5012 nM T29683 C08BLI 25221995 Ki = 0.8 nM T29683 C3VJ0E 25222441 Ki = 3.1 nM T29683 CN82RQ 30127472 IC50 > 10000 nM T29683 C82LDX 31915241 IC50 = 5090 nM T29683 CM28OR 44215995 Ki = 3.981 nM T29683 CD0J1R 44215996 Ki = 7.943 nM T29683 C73ILF 44216236 Ki = 0.91 nM T29683 CHK2D4 44216344 Ki = 20 nM T29683 CO9N0V 44241710 Ki = 0.7 nM T29683 CRQB98 44241723 Ki = 0.2 nM T29683 CP37XK 44266422 Ki = 2.2 nM T29683 C0WK7U 44266459 Ki = 1.2 nM T29683 CYBO34 44266493 Ki = 1.5 nM T29683 CCMW03 44266500 Ki = 1144 nM T29683 C3CPS4 44266510 Ki = 2.4 nM T29683 C61EWH 44266517 Ki = 1653 nM T29683 CQ18SV 44266551 Ki = 5.4 nM T29683 C5Q9SI 44266599 Ki = 2.2 nM T29683 C49QTB 44266600 Ki = 1068 nM T29683 CJY2E8 44266632 Ki = 29.9 nM T29683 CD12NY 44266639 Ki = 30.3 nM T29683 CQ04LU 44276673 IC50 = 6.8 nM T29683 C8YE9F 44276738 IC50 = 2.6 nM T29683 CPC5E6 44276792 IC50 = 127 nM T29683 C5O9BF 44281769 IC50 = 9300 nM T29683 C2VG8B 44288758 IC50 = 10000 nM T29683 CQC6I2 44288896 IC50 = 3300 nM T29683 CR1WZ8 44289197 IC50 = 450 nM T29683 CQ5RI8 44290558 IC50 = 28 nM T29683 CQ9P2K 44290617 IC50 = 39 nM T29683 CJP5E7 44290618 IC50 = 1490 nM T29683 C9XWT1 44290762 IC50 = 18 nM T29683 C53XBO 44290890 IC50 = 8620 nM T29683 CC18ZK 44290902 IC50 = 67 nM T29683 CKA7E3 44290917 IC50 = 5890 nM T29683 C4X1RZ 44290948 IC50 = 9610 nM T29683 CFKB43 44291015 IC50 = 40 nM T29683 CL1T5C 44291016 IC50 = 229 nM T29683 CEB42P 44291084 IC50 = 101 nM T29683 CQ39ZM 44291361 IC50 = 5890 nM T29683 C0IWG5 44291441 IC50 = 1520 nM T29683 C0VNU9 44291442 IC50 = 10000 nM T29683 CH16ID 44291515 IC50 = 39 nM T29683 CD4P2Y 44291545 IC50 = 102 nM T29683 CB13RE 44291546 IC50 = 1690 nM T29683 C93NXY 44291547 IC50 = 425 nM T29683 C7YA0S 44291656 IC50 = 229 nM T29683 CACZ20 44291787 IC50 = 92 nM T29683 CEA5M3 44291788 IC50 = 40 nM T29683 CF52ZM 44294476 IC50 = 1200 nM T29683 CN8UW7 44301357 IC50 = 9420 nM T29683 CHEC65 44308430 EC50 > 10000 nM T29683 CRT79O 44308431 EC50 > 10000 nM T29683 C6ONP4 44308550 EC50 > 10000 nM T29683 CK8W5Q 44308551 EC50 > 10000 nM T29683 C3J6QU 44315209 Ki = 674 nM T29683 CH30NT 44315210 Ki = 572 nM T29683 C9PT3J 44315231 Ki = 312 nM T29683 CM9KT1 44315267 Ki = 103 nM T29683 CKT98C 44315297 Ki = 10.9 nM T29683 CAT8U5 44315298 Ki = 2.2 nM T29683 CF50BD 44315299 Ki = 3.2 nM T29683 CF2EQ0 44315369 Ki = 20 nM T29683 C70HNK 44315370 Ki = 11.8 nM T29683 C4GLI3 44315390 Ki = 11 nM T29683 C1S2MC 44315421 Ki = 304 nM T29683 CCW50R 44315422 Ki = 176 nM T29683 C46IEH 44315483 Ki = 0.3 nM T29683 C6TRV5 44315572 Ki = 97 nM T29683 CS9K4I 44315573 Ki = 231 nM T29683 CHX17S 44315576 Ki = 29 nM T29683 CDX84T 44315589 Ki = 945 nM T29683 C94WGI 44315590 Ki = 281 nM T29683 C0UK2L 44315591 Ki = 167 nM T29683 CY48NV 44346117 IC50 = 10000 nM T29683 C1WQ2A 44359485 EC50 = 0.21 nM T29683 C2S4RW 44418978 IC50 = 2 nM T29683 C93VJL 44418979 IC50 = 3.3 nM T29683 C16FUK 44418980 IC50 = 1.9 nM T29683 CS08LV 44418981 IC50 = 1.6 nM T29683 CP9VN3 44418982 IC50 = 0.72 nM T29683 CS5EY1 44418983 IC50 = 5.7 nM T29683 CHF36T 44418984 IC50 = 1.5 nM T29683 CF1A6T 44418985 IC50 = 3.5 nM T29683 C85GLF 44418986 IC50 = 3.5 nM T29683 CHS73F 44418998 IC50 = 17 nM T29683 C1FM8H 44419014 IC50 = 12 nM T29683 C5MT2W 44419015 IC50 = 5.8 nM T29683 C7GY8W 44419017 IC50 = 51 nM T29683 CW1DP9 44419019 IC50 = 37 nM T29683 C9H0DC 44419033 IC50 = 5.8 nM T29683 C7OI8A 44419059 IC50 = 160 nM T29683 CCY70M 44419061 IC50 = 34 nM T29683 C8PJ6U 44419062 IC50 = 17 nM T29683 C13BLN 44419687 IC50 = 0.85 nM T29683 CLZ8V5 44419691 IC50 = 22 nM T29683 C16EQT 44419696 IC50 = 60 nM T29683 COD6W8 44419703 IC50 = 190 nM T29683 CPFQ78 44419704 IC50 = 91 nM T29683 CRC4J0 44419708 IC50 = 8.4 nM T29683 CSU9T6 44419712 IC50 = 39 nM T29683 C51DKS 44419717 IC50 = 110 nM T29683 C43QJZ 44419718 IC50 = 22 nM T29683 CQOD95 44419721 IC50 = 24 nM T29683 CT37PA 44419722 IC50 = 11 nM T29683 C8E5CW 44419728 IC50 = 38 nM T29683 C1WT4B 44419729 IC50 = 28 nM T29683 CR30LY 44419732 IC50 = 4.1 nM T29683 C3G0CP 44419733 IC50 = 430 nM T29683 CTZ42J 44419759 IC50 = 57 nM T29683 C1H7YR 44444681 IC50 > 3000 nM T29683 CPMZ84 44458598 IC50 > 5000 nM T29683 CX0TU1 44458983 IC50 > 5000 nM T29683 C0GUN2 44459032 IC50 > 5000 nM T29683 C4DL5C 44469677 IC50 > 10000 nM T29683 CG1QT9 44550460 Ki = 10.4 nM T29683 C72FAY 44570858 Ki = 15.85 nM T29683 C47CPI 44570859 Ki = 5.012 nM T29683 CE40QM 44570897 Ki = 251.19 nM T29683 CO78QJ 44570898 Ki = 3.162 nM T29683 CIX2K4 44570899 Ki = 5.012 nM T29683 C4DO6S 44570934 Ki = 6.31 nM T29683 CUV82Y 44570935 Ki = 10 nM T29683 COWP35 44570936 Ki = 1.259 nM T29683 CLA5R8 44570937 Ki = 1.259 nM T29683 CH12DC 44570979 Ki = 6.31 nM T29683 C96TPM 44570980 Ki = 1.585 nM T29683 C63IRV 46889466 Ki = 93.25 nM T29683 CZS8I3 46889667 Ki = 0.95 nM T29683 C91JMT 46889668 Ki = 15.1 nM T29683 C7I4CK 46889669 Ki = 6.87 nM T29683 C9FM0R 46889690 Ki = 8.38 nM T29683 C0FBN7 46889691 Ki = 7.72 nM T29683 CLT23D 46889692 Ki = 29.73 nM T29683 C3VA6U 46889693 Ki = 0.74 nM T29683 C8ZO3Y 46889694 Ki = 7.27 nM T29683 CO39TW 46889695 Ki = 1.48 nM T29683 CPSE79 46889696 Ki = 1.12 nM T29683 CPYO39 46889697 Ki = 29.79 nM T29683 CO1R8E 46889698 Ki = 0.91 nM T29683 C93GXR 51003494 Ki = 7.6 nM T29683 CD2YU8 51351496 IC50 = 180 nM T29683 C2UG4W 51351504 IC50 = 180 nM T29683 CE8J6X 52932923 Ki = 31.62 nM T29683 CYP7K5 52933155 Ki = 5.012 nM T29683 COMU84 52940879 Ki = 298 nM T29683 CBP7R5 52942335 Ki = 5.012 nM T29683 CQX80G 52943089 Ki = 370 nM T29683 C9LF4T 52943090 Ki = 165 nM T29683 CZC98M 52943534 Ki = 3.162 nM T29683 CSY8P6 52943546 Ki = 6.31 nM T29683 C8UN7I 52946726 Ki = 192 nM T29683 C1VQ5F 52947688 Ki = 100 nM T29683 CNB3X5 52947724 Ki = 158.49 nM T29683 C8VL0O 52948404 Ki = 5.012 nM T29683 C1DJ5W 52949416 Ki = 1300 nM T29683 CTYM48 53087371 IC50 = 7200 nM T29683 C7T4MG 53308735 EC50 = 3.7 nM T29683 CX29AL 53317081 Ki = 5.3 nM T29683 CA9T3H 53317082 Ki = 24 nM T29683 CM7ZK1 53317083 Ki = 140 nM T29683 CN2W9V 53317092 Ki = 12 nM T29683 CS36UK 53317093 Ki = 7.8 nM T29683 CIGP04 53317094 Ki = 1.8 nM T29683 C0ZF7Q 53317130 EC50 = 1.8 nM T29683 CA3SQ7 53317131 EC50 = 18 nM T29683 C3UGH5 53317537 EC50 = 110 nM T29683 CYZ24V 53317679 Ki = 1.9 nM T29683 C3UMY8 53317711 Ki = 70 nM T29683 CK9SA5 53318369 Ki = 15 nM T29683 CJ81OE 53318370 Ki = 14 nM T29683 CD1PW0 53318371 Ki = 47 nM T29683 C2Y0GL 53318388 Ki = 3.6 nM T29683 CCWH06 53318389 Ki = 3.3 nM T29683 CE10HM 53318390 Ki = 8.7 nM T29683 CX73VD 53318419 EC50 = 81 nM T29683 CFT35O 53318420 EC50 = 1.8 nM T29683 C68AVO 53318840 EC50 = 15 nM T29683 CWF6U5 53319705 Ki = 33 nM T29683 C8LBF5 53319706 Ki = 23 nM T29683 C8P1UA 53319707 Ki = 1000 nM T29683 CXNV67 53319708 Ki = 210 nM T29683 C3SF4M 53319719 Ki = 2.8 nM T29683 CO2YF0 53319720 Ki = 5.8 nM T29683 C7B3GQ 53320155 EC50 = 38 nM T29683 CLX75C 53320156 EC50 = 74 nM T29683 C7N1TM 53320999 Ki = 18 nM T29683 CV3YZ5 53321000 Ki = 50 nM T29683 CN30ZS 53321001 Ki = 5.8 nM T29683 C8ZVO5 53321002 Ki = 56 nM T29683 CXC8D3 53321008 Ki = 5.6 nM T29683 CI8DY1 53321470 EC50 = 8.2 nM T29683 C8HG6X 53321471 EC50 = 3.6 nM T29683 CI0T6Y 53321639 Ki = 28 nM T29683 CTI8Z6 53321640 Ki = 270 nM T29683 CG01LF 53322346 Ki = 13 nM T29683 CJX3B8 53322347 Ki = 110 nM T29683 CT71IZ 53322353 Ki = 1.5 nM T29683 CE5GA2 53322354 Ki = 150 nM T29683 CU82JN 53322390 EC50 = 5.3 nM T29683 C8YCW6 53322796 EC50 = 1900 nM T29683 CHM79E 53322797 EC50 = 5.1 nM T29683 C08EUT 53322798 EC50 = 77 nM T29683 CT0M8Q 53323699 Ki = 16 nM T29683 CTHX67 53323700 Ki = 5.9 nM T29683 CPU84K 53323701 Ki = 32 nM T29683 CI6A9N 53323702 Ki = 140 nM T29683 CAO86S 53323703 Ki = 32 nM T29683 CPTY26 53323714 Ki = 3.7 nM T29683 CRP7D0 53323715 Ki = 17 nM T29683 CS4WT0 53323716 Ki = 12 nM T29683 CB3K2L 53323748 EC50 = 1.7 nM T29683 CTV27A 53323749 EC50 = 16 nM T29683 CXJ09K 53324128 EC50 = 13 nM T29683 C78HOZ 53324284 Ki = 11 nM T29683 C37RTW 53324972 Ki = 4.6 nM T29683 CXR48D 53324973 Ki = 67 nM T29683 C6SYC7 53324974 Ki = 37 nM T29683 CMS2O1 53324975 Ki = 40 nM T29683 C7NS6W 53324976 Ki = 7.3 nM T29683 CG7PR6 53324988 Ki = 7.3 nM T29683 CDBK64 53325015 EC50 = 2500 nM T29683 C9VE8J 53325016 EC50 = 12 nM T29683 CB3IK1 53325403 EC50 = 3.3 nM T29683 CK18CL 53325439 EC50 = 212 nM T29683 C5LFA4 53325440 EC50 = 38 nM T29683 C3JK6Y 53325441 EC50 > 9300 nM T29683 CWT67H 53325566 Ki = 1900 nM T29683 CZA14B 53325578 EC50 = 1120 nM T29683 CWJ2D3 53326273 Ki = 12 nM T29683 C4GLU5 53326274 Ki = 67 nM T29683 C6Q0DB 53326275 Ki = 350 nM T29683 CQ08ZU 53326280 Ki = 140 nM T29683 C51VSL 53326315 EC50 = 48 nM T29683 CFC6D2 53326316 EC50 = 690 nM T29683 CI8H0G 53326317 EC50 = 220 nM T29683 C9OI2E 53326646 Ki = 93 nM T29683 CU08CK 53326688 EC50 = 7.7 nM T29683 C24RZJ 53326689 EC50 = 88 nM T29683 CX2AI0 53326690 EC50 = 16 nM T29683 CP45OS 53326864 Ki = 14 nM T29683 CY0E9L 53326884 Ki = 24 nM T29683 C92IXZ 53326885 Ki = 90 nM T29683 CDL78Q 53326891 Ki = 7.5 nM T29683 CK1C9O 53472113 Ki = 1.995 nM T29683 C2W0ZI 53482149 Ki = 501.19 nM T29683 C9EF7S 53482945 IC50 = 4000 nM T29683 CA9G0H 53482947 Ki = 1584.89 nM T29683 CQU40H 53482949 Ki = 1258.93 nM T29683 COR86Y 54579946 IC50 = 190 nM T29683 CBX31W 54579947 IC50 = 93 nM T29683 C5SBF2 54579948 IC50 = 2000 nM T29683 C5CTZ3 54579949 IC50 = 1300 nM T29683 CD9OY4 54580928 IC50 = 42 nM T29683 CCX80E 54580929 IC50 = 2900 nM T29683 CL7S5M 54580930 IC50 = 3100 nM T29683 COIH43 54580975 IC50 = 370 nM T29683 C1VLY8 54582921 IC50 > 5000 nM T29683 C1KHI9 54582922 IC50 = 2500 nM T29683 CLVU42 54582923 IC50 = 7100 nM T29683 CQV37E 54582966 Ki = 20 nM T29683 CK6G9H 54582967 IC50 > 10000 nM T29683 CA52PI 54582968 IC50 > 10000 nM T29683 C9NP0K 54583920 IC50 = 7400 nM T29683 CFDT72 54583921 IC50 = 205 nM T29683 C3QZY5 54583958 IC50 = 3300 nM T29683 CEFT05 54583959 IC50 = 130 nM T29683 CT7QE3 54584864 IC50 = 480 nM T29683 CILC50 54584865 IC50 = 280 nM T29683 C04AQE 54584866 IC50 > 10000 nM T29683 C1W5FQ 54584909 IC50 = 1200 nM T29683 CZ4RQ7 54584910 IC50 = 580 nM T29683 CSX41C 54584911 IC50 = 180 nM T29683 CXL2Z3 54585832 IC50 = 208 nM T29683 CVC2N7 54585869 IC50 = 1800 nM T29683 CUM85L 54585870 IC50 > 10000 nM T29683 CF8MY7 54586801 IC50 = 3100 nM T29683 C7OX8S 54586802 IC50 = 130 nM T29683 C2P9FH 54586837 IC50 = 80 nM T29683 C53NEF 57392804 Ki = 1.585 nM T29683 C3I2PJ 57396275 Ki = 5.012 nM T29683 CTY0J1 57398076 Ki = 1.995 nM T29683 C10WAF 57403249 Ki = 1 nM T29683 C4S3FE 67450880 IC50 = 15.85 nM T29683 C18YOM 67452275 IC50 = 260 nM T29683 CDR4T8 67452845 IC50 = 1584.89 nM T29683 CQ1D4M 67453148 Ki = 794.33 nM T29683 C8L5HO 67453320 Ki = 501.19 nM T29683 CWY7B2 67455077 Ki = 7943.28 nM T29683 CKZH35 67970499 Ki > 31622.78 nM T29683 C62ULC 71225056 Ki = 398.11 nM T29683 C7PK5T 71452185 Ki = 0.6 nM T29683 C71KGJ 71453994 Ki = 2.5 nM T29683 CQ82SD 71455736 Ki = 1 nM T29683 CC1XL3 71457524 Ki = 0.6 nM T29683 CN8CM1 71533722 Ki = 12.59 nM T29683 CKB12X 71549359 Ki = 79.43 nM T29683 C4LZM6 71549637 Ki = 6.31 nM T29683 C6JOB5 71549767 Ki = 25.12 nM T29683 CV47CJ 71549769 Ki = 3.162 nM T29683 C5IV9D 71549913 Ki = 10 nM T29683 CRE34C 71582890 EC50 = 0.11 nM T29683 CPZ01Q 71582891 EC50 = 0.15 nM T29683 C24WPK 71583209 EC50 = 0.04 nM T29683 C53OMK 71583210 EC50 = 0.024 nM T29683 C3OU1J 71583328 EC50 = 0.08 nM T29683 C38KLS 71583329 EC50 = 0.026 nM T29683 CZ9L3G 71583445 EC50 = 0.017 nM T29683 CKN09M 71583446 EC50 = 0.072 nM T29683 CS2RU3 71583561 EC50 = 0.28 nM T29683 CV46NK 71583562 EC50 = 0.065 nM T29683 CYA26E 71583665 EC50 = 0.051 nM T29683 CH45FA 71583666 EC50 = 0.06 nM T29683 CZ39PR 71583776 EC50 = 0.012 nM T29683 CX29ZY 71583777 EC50 = 0.036 nM T29683 C5SGQ3 71583894 EC50 = 0.043 nM T29683 C5GS4K 71583895 EC50 = 0.04 nM T29683 C43WRS 71583996 EC50 = 0.046 nM T29683 C5I1KL 71583997 EC50 = 0.032 nM T29683 C6FDT7 71584103 EC50 = 0.041 nM T29683 CZA9D2 71584104 EC50 = 0.036 nM T29683 CRB8F0 71584221 EC50 = 0.083 nM T29683 CCVD30 71584355 EC50 = 0.078 nM T29683 CZRL61 71584356 EC50 = 0.0054 nM T29683 CO6T9B 71584479 EC50 = 0.071 nM T29683 C0XN3T 71584480 EC50 = 0.085 nM T29683 CKQ56I 71584609 EC50 = 0.47 nM T29683 C8EVK7 71716520 EC50 = 0.038 nM T29683 C9DFV6 71717757 EC50 = 0.12 nM T29683 CPIO21 71718360 EC50 = 5.04 nM T29683 CQX9U5 71720166 EC50 = 1.38 nM T29683 C30MKX 71720167 EC50 = 0.13 nM T29683 CWH6T3 72548703 IC50 = 8.2 nM T29683 CP5HC1 73212363 Ki > 10000 nM T29683 C86LGQ 73212437 Ki = 10000 nM T29683 C6DXY3 73212439 Ki = 1000 nM T29683 C83GFJ 73212440 Ki = 10000 nM T29683 CR36KA 73212441 Ki > 10000 nM T29683 C1Y6IU 73212515 Ki = 10000 nM T29683 CA64UI 73212516 Ki > 10000 nM T29683 CFC47O 73212517 Ki = 10000 nM T29683 CG9JP6 73212518 Ki = 10000 nM T29683 CU30GO 73212519 Ki = 10000 nM T29683 CE9R0Y 73212588 Ki > 10000 nM T29683 CEU1C3 73212589 Ki > 10000 nM T29683 CKT46G 73212590 Ki = 10000 nM T29683 C7Q1UP 73212591 Ki > 10000 nM T29683 CGU23K 73212592 Ki > 10000 nM T29683 C0K4EH 73212593 Ki > 10000 nM T29683 CG4J9A 73350299 IC50 = 112 nM T29683 CCN15O 73351568 EC50 = 3.36 nM T29683 C6EB5R 73775687 IC50 = 22 nM T29683 CH73SX 73775808 IC50 = 43 nM T29683 CAV2B0 73775809 EC50 = 91 nM T29683 C6S4TN 73775940 EC50 = 240 nM T29683 C51RPE 73775941 EC50 = 350 nM T29683 CB45FG 76317390 Ki = 72.44 nM T29683 C9GQS2 81689815 Ki = 100 nM T29683 C4T3IW 86272102 IC50 = 6.31 nM T29683 C13AJC 86274362 Ki = 100 nM T29683 C3OLB1 86274489 Ki = 19.95 nM T29683 CAB78T 86274732 Ki = 31.62 nM T29683 CCU13T 86275207 Ki = 50.12 nM T29683 CJ68CO 86275449 Ki = 125.89 nM T29683 CW01SX 90417750 Ki = 316.23 nM T29683 CD5W6K 90417914 Ki = 3.162 nM T29683 C7E2NA 90644603 Ki = 1584.89 nM T29683 CGYH84 90644605 Ki = 1258.93 nM T29683 CU3KJ2 90644607 Ki = 3981.07 nM T29683 C6OXD3 90644609 Ki = 6309.57 nM T29683 C5OXI0 90644611 Ki = 2511.89 nM T29683 CI0P4O 90644613 Ki = 63.1 nM T29683 CN3EA2 90644615 Ki = 10000 nM T29683 CQ84WX 90644617 Ki = 1995.26 nM T29683 C5D2IJ 90644619 Ki = 50.12 nM T29683 CW2LI9 90644621 Ki = 1584.89 nM T29683 C8O9CH 90644623 Ki = 39.81 nM T29683 C13NEK 90644625 Ki = 794.33 nM T29683 CI46TV 90644627 Ki = 19.95 nM T29683 CGR64B 90644629 Ki = 31.62 nM T29683 CTQD75 90644630 Ki = 1000 nM T29683 C4UYZ6 90644631 Ki = 2.512 nM T29683 C1GRO9 90644632 Ki = 125.89 nM T29683 C2CRO1 90644633 Ki = 7.943 nM T29683 C58BJM 90644634 Ki = 25.12 nM T29683 CYF4L3 90663905 IC50 = 1760 nM T29683 CZ17TH 90663907 IC50 = 3270 nM T29683 CJ06SU 91535935 IC50 = 8 nM T29683 C9ZUP4 91809194 EC50 = 0.041 nM T29683 CNS4V9 102531123 EC50 = 0.064 nM T29683 CXL57K 102531124 EC50 = 0.05 nM T29683 CY8R0C 102531125 EC50 = 0.03 nM T29683 C0OSW4 102531127 EC50 = 0.019 nM T29683 C8F6VO 117604931 IC50 = 19.95 nM T29683 C2MFX8 118724962 EC50 > 100000 nM T29683 C2I9WR 118724963 EC50 > 100000 nM T29683 CK6VT5 118724964 EC50 = 16 nM T29683 C3U2HT 118724965 EC50 = 920 nM T29683 CFQ6V5 118724966 EC50 = 1900 nM T29683 C92MQV 118724967 EC50 = 370 nM T29683 CJ0N7O 118724968 EC50 = 100 nM T29683 C0SM3L 118735340 Ki = 76 nM T29683 C8MQ9Z 118735341 Ki > 31622.78 nM T29683 C4N3PG 118735342 Ki = 5011.87 nM T29683 CI69BV 118735343 Ki > 31622.78 nM T29683 CB8CE2 118735344 Ki > 31622.78 nM T29683 CAX5Q0 118735345 IC50 = 3981.07 nM T29683 C1WG6O 118735346 Ki > 31622.78 nM T29683 C1TOB9 118735347 Ki > 31622.78 nM T29683 C7Z9PQ 118735348 IC50 = 10000 nM T29683 C86YDG 118735349 Ki = 63.1 nM T29683 C0T9KC 118735350 Ki = 1584.89 nM T29683 C7WTU3 118735351 Ki = 6309.57 nM T29683 C8A2HI 118735352 Ki > 31622.78 nM T29683 CAN90V 118735353 Ki = 12.59 nM T29683 C4XY9I 118735354 IC50 = 63.1 nM T29683 C1XL4S 118735355 Ki = 2.512 nM T29683 CSP7R8 122187066 Ki = 10000 nM T29683 CQA8B2 122187067 Ki = 25.12 nM T29683 C3ZA9G 122187068 Ki = 1258.93 nM T29683 CS5CF1 122187069 Ki = 199.53 nM T29683 C76XAE 125111645 EC50 = 0.029 nM T29683 CO4N2F 127034660 EC50 = 0.018 nM T29683 CNQ2Y4 127034696 EC50 = 0.012 nM T29683 CRAC83 127034748 EC50 = 0.022 nM T29683 CV9Z2G 127034749 EC50 = 0.0091 nM T29683 CJ7T9U 127034767 EC50 = 0.006 nM T29683 CE9Z2Y 127034768 EC50 = 0.0029 nM T29683 C7CYF5 127034769 EC50 = 0.011 nM T29683 CNX2F4 127034928 EC50 = 0.014 nM T29683 CATQ52 127034940 EC50 = 0.0074 nM T29683 CL6OW2 127035038 EC50 = 0.024 nM T29683 C1AG9R 127035039 EC50 = 0.0081 nM T29683 C8WXA7 127035040 EC50 = 0.018 nM T29683 CE62OX 127035105 EC50 = 0.013 nM T29683 CHAS82 127035106 EC50 = 0.043 nM T29683 CJR2D5 127035222 EC50 = 0.017 nM T29683 C29BAM 127035348 IC50 > 10000 nM T29683 C52ALH 127035367 EC50 = 0.084 nM T29683 C2S8IW 127035368 EC50 = 0.083 nM T29683 CR82NL 127035511 IC50 > 10000 nM T29683 CUV12X 127035512 EC50 = 0.031 nM T29683 C9PDL3 127035576 EC50 = 0.0025 nM T29683 CS78HG 127035706 EC50 = 0.033 nM T29683 C1N5JV 127035707 IC50 > 10000 nM T29683 C2PL6V 127036728 EC50 = 0.017 nM T29683 CO4VJ5 127048298 IC50 = 44 nM T29683 C2RB3Q 127049013 IC50 = 24 nM T29683 CZ7J2Q 127049014 IC50 = 5.6 nM T29683 CK1S3I 127049297 IC50 = 1527 nM T29683 CI6V3K 127049298 IC50 = 965 nM T29683 CAM3Z5 127052434 IC50 = 154 nM T29683 CNTC08 127052725 IC50 > 10000 nM T29683 C9S4AD 127052726 IC50 > 10000 nM T29683 CX6U7K 135406470 Ki = 493 nM T29683 C19PZJ 135419384 Ki = 653 nM T29683 C1JKC0 135430775 IC50 > 1000 nM T29683 C1Y3IB 135449286 IC50 = 150 nM T29683 CJVK41 136094788 IC50 = 3.9 nM T29683 C3B5AN 136094789 IC50 = 245 nM T29683 CQ95FP 136094790 IC50 = 390 nM T29683 CCQ2R7 136094791 IC50 = 6 nM T29683 CTD69B 137647980 IC50 = 2500 nM T29683 CQ4ZE2 145864510 IC50 = 10300 nM T29683 C7UNL0 145864511 IC50 = 8200 nM T29683 CE4MY6 145864512 IC50 = 4100 nM T29683 C4PK2Y 155512473 IC50 = 11800 nM T29683 CN7T3Z 155540643 IC50 = 13700 nM T29683 C72EFN 155551678 Ki = 0.3 nM T29683 D00HUY 10473960 IC50 > 5000 nM T29683 D01NPA 5311311 EC50 = 53 nM T29683 D02CCA 25195091 Ki = 10 nM T29683 D04TXE 5311350 IC50 = 40 nM T29683 D07NNN 5311312 Ki = 0.7943 nM T29683 D09NBN 9915428 IC50 = 7 nM T29683 D0G2AK 44419758 IC50 = 32 nM T29683 D0J3AO 9914897 IC50 = 16 nM T29683 D0J8SU 36511 EC50 = 793 nM T29683 D0O8RG 2849628 IC50 = 33.5 nM T29683 D0S9CI 11989776 IC50 = 3 nM T29683 D0U9IB 10328936 EC50 = 0.22 nM T29683 D0W3XD 16049828 IC50 = 4.5 nM T29683 D0Z6TG 9852253 Ki = 74 nM T62410 C7ECX6 5387164 IC50 = 4797.33 nM T62410 C2KZF0 5476176 IC50 = 5997.91 nM T62410 CUWD62 5712167 IC50 = 3800 nM T62410 CZP2V5 5712224 IC50 = 9506.05 nM T62410 C0SKR3 5775365 IC50 = 510 nM T62410 CQ32GK 5839766 IC50 = 10000 nM T62410 CN9OX4 5929655 IC50 = 7700 nM T62410 CD0CI2 6035979 IC50 = 11994.99 nM T62410 CN47BA 8826735 IC50 = 2090 nM T62410 CB3L8H 8832830 IC50 = 5000 nM T62410 CBPY06 8832834 IC50 = 10000 nM T62410 CBVC52 8854038 IC50 = 2700 nM T62410 CH8D5Q 8858338 IC50 = 359.75 nM T62410 C6UX4J 10633725 IC50 = 12000 nM T62410 CPX74Q 10662259 IC50 = 11100 nM T62410 C5CA1S 10759357 IC50 = 899.5 nM T62410 C37TVX 10760359 IC50 = 2460.37 nM T62410 CD97WY 10780801 IC50 = 1900 nM T62410 C8BV5Y 11043793 IC50 = 1399.59 nM T62410 CNTJ13 11054705 IC50 = 1698.24 nM T62410 C2HFY3 19553304 IC50 = 3900 nM T62410 CYI18V 19561174 IC50 = 5000 nM T62410 C20ZDI 19562959 IC50 = 749.89 nM T62410 CJ5ED8 44301768 IC50 = 749.89 nM T62410 CS5UK8 44516427 IC50 = 1180 nM T62410 C0LVG5 45257601 IC50 = 3300 nM T62410 C6F4RU 76311813 IC50 = 709.58 nM T62410 CXU9F5 76311814 IC50 = 799.83 nM T62410 CYEO36 76311815 IC50 = 1140.25 nM T62410 CQZ73X 76315377 IC50 = 4295.36 nM T62410 CYB74V 76315388 IC50 = 4602.57 nM T62410 C3XS8B 76319043 IC50 = 2300 nM T62410 C3OP2B 76319044 IC50 = 3198.9 nM T62410 CUW94I 76319065 IC50 = 2798.98 nM T62410 CZ84DQ 76322700 IC50 = 920 nM T62410 CNU98S 76326279 IC50 = 3097.42 nM T62410 C7ZGX3 76329888 IC50 = 1380 nM T62410 CXWR38 76333525 IC50 = 770 nM T62410 C4DV1O 76333526 IC50 = 1000 nM T62410 C5H3CO 76333527 IC50 = 1000 nM T62410 CDEG91 76333528 IC50 = 5794.29 nM T62410 CT0F3U 76333529 IC50 = 230.14 nM T89918 D0SV8E 126941 IC50 > 20000 nM T89918 D0Y4GO 135410875 IC50 = 11.74 nM T89918 D06YIB 135436405 IC50 = 220 nM T89918 C7OTP8 3439 IC50 > 30000 nM T89918 CF1M8Q 468708 IC50 > 30000 nM T89918 CHKA59 11963491 Ki > 100000 nM T89918 CHB34X 11963492 Ki = 4800 nM T89918 CBU8F6 12413165 Ki > 100000 nM T89918 CTA8R7 24748572 IC50 = 13.8 nM T89918 C7O3JT 24771725 IC50 = 13.3 nM T89918 C07HBN 24771726 IC50 = 23.6 nM T89918 CLF6B9 42637226 IC50 = 32.3 nM T89918 C3SMD7 42637584 IC50 = 26.6 nM T89918 CPM3L5 67092576 IC50 = 82 nM T89918 CTK64O 67092918 IC50 = 101 nM T89918 C9EA3J 135407589 IC50 = 3000 nM T89918 CUS5Q1 135413518 IC50 = 5.77 nM T89918 C5LDN0 135455947 IC50 = 5300 nM T89918 CV46BA 135465343 Ki = 130 nM T89918 CV47OY 135474781 Ki = 15 nM T89918 C20PSX 135483994 Ki = 35 nM T89918 C79OVQ 135488791 Ki = 4000 nM T89918 C2R9FW 135491785 Ki = 5000 nM T89918 C95DCY 135493624 Ki = 38 nM T89918 CEW67A 135497378 Ki = 30 nM T89918 C35JUA 135501119 Ki = 14 nM T89918 CVH8Q5 135502217 IC50 > 20000 nM T89918 CHD01N 135513031 Ki = 21000 nM T89918 C46NSF 135515218 Ki = 32 nM T89918 CP0K9Y 135515593 Ki = 28 nM T89918 C2K0FD 135518696 Ki = 30000 nM T89918 CP0J1I 135529975 Ki = 825 nM T89918 CC7PW9 135548219 Ki = 8.5 nM T89918 CL2AG7 135566721 Ki = 180 nM T89918 CRA6Z7 135566722 Ki = 210 nM T89918 C9Z4ES 135567027 IC50 <= 3 nM T89918 C14LTO 135567028 IC50 = 3.13 nM T89918 CF39AI 135567029 IC50 = 1.8 nM T89918 C8N7ES 135567030 IC50 = 0.6 nM T89918 CGM2V5 135567031 IC50 = 2.03 nM T89918 CTI9E3 135567032 IC50 = 2.89 nM T89918 C94CNA 135567033 IC50 = 5.49 nM T89918 CFE2O7 135567034 IC50 = 1 nM T89918 C8KVP5 135567035 IC50 = 2.6 nM T89918 CSQX75 135567163 IC50 = 2.64 nM T89918 C45BZH 135596568 IC50 = 2060 nM T89918 CTXM18 135596569 IC50 = 140 nM T89918 C0X1QM 135616220 IC50 = 18200 nM T89918 CL74ZW 135616221 IC50 = 4300 nM T89918 C7HAY6 135616222 IC50 = 7600 nM T89918 CIC3S1 135625317 IC50 = 16.2 nM T89918 CMZ27I 135745092 IC50 = 7.2 nM T89918 C06IDH 135746097 IC50 > 17000 nM T89918 C1YVM0 135758974 IC50 = 2600 nM T89918 CQF8P5 135800109 IC50 = 1 nM T89918 C71OSY 135816670 IC50 = 3500 nM T89918 C53HOX 135816671 IC50 = 6600 nM T89918 CV5S7G 135816672 IC50 = 6100 nM T89918 C8NVR1 135816673 IC50 = 3100 nM T89918 CA6ZN8 135816674 IC50 = 18700 nM T89918 C6XK3M 135862924 IC50 = 7650 nM T89918 CY2J7Z 135881773 IC50 > 100000 nM T89918 C0Y2ZJ 135884476 Ki = 14 nM T89918 CWL71S 135887124 IC50 = 4800 nM T89918 CH1W2S 135887126 IC50 = 85900 nM T89918 C6U0PF 135887127 IC50 > 100000 nM T89918 COA6S0 135887128 IC50 > 100000 nM T89918 CFIG79 135887147 IC50 = 5300 nM T89918 CDA05G 135887148 IC50 = 26000 nM T89918 CY1M8B 135924031 IC50 = 8.6 nM T89918 CLBO26 135924167 Ki = 1400 nM T89918 C8R1PU 135924168 Ki = 1100 nM T89918 CN7B0Z 135924169 Ki = 850 nM T89918 CYI9Q7 135924170 Ki = 1100 nM T89918 C5JDL6 135924171 Ki = 1200 nM T89918 CZ5CY0 136002156 IC50 = 52000 nM T89918 C7R8XM 136002207 Ki = 35000 nM T89918 C2SI7N 136002209 Ki > 100000 nM T89918 CRYC07 136002210 Ki = 45000 nM T89918 CE10FO 136026553 Ki = 82100 nM T89918 CI4HM6 136035744 Ki = 15 nM T89918 CU1T3Q 136035745 Ki = 2 nM T89918 CF60KR 136035746 Ki = 3.4 nM T89918 CTD67N 136035747 Ki = 3 nM T89918 C7BNR9 136035748 Ki = 35 nM T89918 CVM94X 136035749 Ki = 2000 nM T89918 C6HL7E 136044121 IC50 > 40000 nM T89918 C76AYL 136044122 IC50 > 20000 nM T89918 C6F9VM 136044123 IC50 > 20000 nM T89918 CD37LT 136044139 Ki = 1300 nM T89918 CR7UY3 136044173 IC50 = 12 nM T89918 C7B9XC 136045806 IC50 > 1000 nM T89918 CK8U2L 136056477 IC50 > 20000 nM T89918 C64VHT 136056601 IC50 > 25000 nM T89918 CNTJ30 136056602 IC50 = 0.00005 nM T89918 CLFS31 136056603 IC50 = 0.0011 nM T89918 C1M8FU 136056604 IC50 = 0.001 nM T89918 CTD19V 136056605 IC50 > 20000 nM T89918 CVY71E 136056606 IC50 = 0.00055 nM T89918 CZG8W6 136059167 IC50 = 1.8 nM T89918 CZC95Y 136059168 IC50 = 4.8 nM T89918 C0C2SJ 136152907 Ki = 1800 nM T89918 CNDZ46 136152908 Ki = 600 nM T89918 CW6Y0D 136152909 Ki > 100000 nM T89918 C4Q1HF 136180345 IC50 = 61.03 nM T89918 CVOC10 136241611 IC50 = 9.62 nM T89918 CMKA64 155517044 IC50 = 5.58 nM T89918 CCL3Y9 155518053 IC50 = 1.2 nM T89918 C91SVN 155519837 IC50 = 6.62 nM T89918 CT70WU 155530762 IC50 = 0.7 nM T89918 CX42MF 155532591 IC50 = 5.25 nM T89918 CFU98A 155534971 IC50 = 2.11 nM T89918 C6S7OC 155548982 IC50 = 1 nM T89918 CX3K8F 155549935 IC50 <= 3 nM T89918 CJ0MK5 155554671 IC50 = 2 nM T89918 CYQ0I9 155555353 IC50 = 4.95 nM T89918 C9FKS7 9910387 Ki = 186000 nM T89918 D0F2WA 135929093 Ki = 30 nM T89918 D0R7LQ 135884475 IC50 = 1600 nM T89918 D0Z9QC 135517463 Ki = 2000 nM T03687 D0E3SH 6918837 Ki = 1.2 nM T03687 D0E7PQ 5311 IC50 = 38 nM T03687 D0L7LC 5352062 Ki = 1100 nM T03687 D0Y3KG 3121 IC50 > 2000000 nM T03687 D05KED 53340666 IC50 > 10000 nM T03687 D07FPY 6918877 Ki = 19 nM T03687 D09XIZ 11538455 Ki = 3.8 nM T03687 D0B1FE 3194 IC50 = 3700 nM T03687 D0B3FV 6445533 IC50 = 8.24 nM T03687 D0B7CH 4775 IC50 > 2000000 nM T03687 D0E6UZ 54575456 IC50 = 554 nM T03687 D0GH3Q 9804992 Ki = 390 nM T03687 D0L2UQ 49855250 Ki = 24 nM T03687 D0M8FD 4261 IC50 > 1000 nM T03687 D0XT6W 6918638 Ki = 24 nM T03687 D0Z4RC 24756910 IC50 = 67.2 nM T03687 D0J8OC 5186 IC50 = 700 nM T03687 D0L1NO 72722126 IC50 = 60 nM T03687 D0QX3G 71532921 IC50 > 10000 nM T03687 D0YN2T 86302836 IC50 = 30 nM T03687 CBIR94 10313 IC50 > 33330 nM T03687 C1N2KZ 88129 IC50 = 91000 nM T03687 C35INR 338818 IC50 = 7840 nM T03687 CH1JD3 419176 IC50 > 2000000 nM T03687 CU3HS2 1108280 IC50 > 100000 nM T03687 C18ENP 6918846 Ki = 24 nM T03687 CC0EU7 9828788 IC50 > 10000 nM T03687 C81EYJ 9923508 IC50 = 3.9 nM T03687 CQG4V8 9924543 IC50 = 2.3 nM T03687 C7RC1E 10309899 IC50 = 28 nM T03687 CG9L1R 10435243 IC50 = 1024 nM T03687 C60QVT 10460379 IC50 = 2344 nM T03687 CG9OC4 11682502 IC50 = 40.7 nM T03687 CYB26W 11688197 IC50 > 1000 nM T03687 C9G1BN 11993595 IC50 = 3300 nM T03687 CH5JS7 11993694 IC50 = 340 nM T03687 C06UTF 13507024 IC50 = 5100 nM T03687 C2D1KP 15983982 Ki = 11 nM T03687 CHB82E 15986417 IC50 = 41400 nM T03687 C52EVH 15986418 IC50 = 8920 nM T03687 CS1QO9 15986509 IC50 = 39300 nM T03687 CFK8J5 16068056 Ki = 11 nM T03687 CMQP70 16068495 Ki = 30 nM T03687 CT84XO 16068594 Ki = 16 nM T03687 CF3ZG5 16068595 Ki = 14 nM T03687 CL60CA 16068912 Ki = 4.4 nM T03687 C17GDO 24779722 IC50 = 247 nM T03687 CY12VH 24825455 Ki = 6100 nM T03687 CX69SY 25066355 IC50 = 1900 nM T03687 CF8VP4 25066356 IC50 = 687 nM T03687 CS9XH7 25066547 IC50 = 1040 nM T03687 C46AGN 25066548 IC50 = 99.6 nM T03687 CJF2M7 25066549 IC50 = 336 nM T03687 CCD5M7 25227504 IC50 = 60.6 nM T03687 CK0D5S 25227505 IC50 = 302 nM T03687 CN97JP 25227508 IC50 = 123 nM T03687 CW8R1B 25227513 IC50 = 322 nM T03687 C43BHY 25269097 IC50 = 927 nM T03687 C2LES7 42599455 IC50 = 4.2 nM T03687 C2KO0F 42599456 IC50 = 2.8 nM T03687 CDT65Y 42631047 IC50 > 100000 nM T03687 CO57GS 44138033 IC50 = 6430 nM T03687 C7F8YJ 44543715 Ki = 10000 nM T03687 CEM91G 44562802 IC50 = 20 nM T03687 CIO34V 44564642 Ki = 21 nM T03687 CA6Q9Y 44592060 IC50 = 11200 nM T03687 C5H8RA 44598536 IC50 > 10000 nM T03687 CSM1O6 45271073 IC50 = 50000 nM T03687 CPSI47 46890583 Ki = 6 nM T03687 C90NYX 46896338 IC50 = 16000 nM T03687 C4DL0M 49847150 IC50 = 5580 nM T03687 CC7Y9U 49850262 IC50 = 621 nM T03687 CI68XL 52912223 IC50 > 100000 nM T03687 C78GKN 53361474 IC50 = 704 nM T03687 CNB63X 53361475 IC50 = 37.8 nM T03687 CQ43VH 53363518 Ki = 5.7 nM T03687 C6Y2EV 53374826 IC50 > 100000 nM T03687 CYQV72 54030066 IC50 = 120 nM T03687 C5A7MU 54613496 IC50 = 1.1 nM T03687 C7OJ4K 56602459 IC50 > 50000 nM T03687 CSY2L7 56602461 IC50 = 12000 nM T03687 CIO96M 56659403 IC50 > 100000 nM T03687 CL18NI 56666337 IC50 > 100000 nM T03687 C9LC5Y 56673234 IC50 > 100000 nM T03687 CWH5N4 56673261 IC50 > 100000 nM T03687 C0ZJG3 56676500 IC50 > 50000 nM T03687 CFUT54 56682413 IC50 = 30000 nM T03687 CZ25SN 56935695 IC50 > 30000 nM T03687 C4LI0D 57521296 IC50 = 50 nM T03687 C1MB4Q 59323957 IC50 > 30000 nM T03687 CK6LX0 59454220 IC50 = 43000 nM T03687 C2SDN1 59454252 IC50 = 13000 nM T03687 CO6A2S 59585196 IC50 = 47000 nM T03687 CPZ5Q3 60148646 IC50 = 790 nM T03687 CP2HK9 60148667 IC50 = 260 nM T03687 C8ZL3J 60148690 IC50 = 80 nM T03687 CK5N4E 60148693 IC50 = 40 nM T03687 C27DKW 60148711 IC50 = 190 nM T03687 CS2E6C 60148712 IC50 = 370 nM T03687 CPF50R 60148997 IC50 = 1800 nM T03687 CB7X2E 60151224 IC50 > 10000 nM T03687 CY05OU 60151225 IC50 > 10000 nM T03687 CWO8H0 60152596 IC50 > 10000 nM T03687 CBN3L0 69950064 Ki = 8 nM T03687 CQY1I6 70789579 Ki = 5980 nM T03687 C7RUE6 71540743 IC50 = 63200 nM T03687 C9LA4F 71540744 IC50 = 32000 nM T03687 C0EK5J 71540745 IC50 > 100000 nM T03687 C80HZX 71540746 IC50 = 34600 nM T03687 C5UZQ0 71540747 IC50 = 18400 nM T03687 C4G5US 71540862 IC50 = 16200 nM T03687 CKR6U8 71583101 IC50 = 800 nM T03687 CBZ5S9 71583103 IC50 = 300 nM T03687 C3PSJ9 71583105 IC50 = 500 nM T03687 C7HG0K 71655802 IC50 > 33330 nM T03687 CPJ4V7 71680913 IC50 > 33000 nM T03687 CI9G3B 71681069 IC50 = 12000 nM T03687 CFUC24 71722010 IC50 > 10000 nM T03687 CI9H6L 72164895 IC50 = 28020 nM T03687 CS5UL7 72195322 IC50 = 48900 nM T03687 CV09DJ 72734543 IC50 = 5000 nM T03687 CM6H9C 76324878 IC50 = 30 nM T03687 CKI74A 76853213 IC50 > 20000 nM T03687 CJ6Z0X 78324068 IC50 > 20000 nM T03687 C3U0KE 81689842 IC50 = 50 nM T03687 CG5ZD9 86291495 IC50 = 5.2 nM T03687 C61VCD 86294741 IC50 = 58000 nM T03687 CBWV30 86294747 IC50 = 34000 nM T03687 CGF12C 86302517 IC50 = 78 nM T03687 C8O5PZ 86302518 IC50 = 57 nM T03687 CL78UP 86302519 IC50 = 42 nM T03687 CY5Q0E 86302520 IC50 = 62 nM T03687 C3EM7H 86581004 IC50 = 35 nM T03687 C7UK3Y 86581005 IC50 = 39 nM T03687 CY64UM 86581152 IC50 = 25 nM T03687 CY5V7C 86581153 IC50 = 45 nM T03687 C1HE8I 86581432 IC50 = 570 nM T03687 CZM07I 86581434 IC50 = 37 nM T03687 C8ZQG9 86581435 IC50 = 50 nM T03687 C6M9PL 86765212 IC50 = 5340 nM T03687 CS5I4Y 87261507 IC50 = 160 nM T03687 CYW51P 90654946 IC50 = 42300 nM T03687 CJH1S6 90654947 IC50 > 100000 nM T03687 CSDO81 90664458 Ki = 24 nM T03687 C0RX4B 90667452 IC50 = 34890 nM T03687 C8HL5V 90667453 IC50 = 61660 nM T03687 C3IE7F 90667454 IC50 = 930 nM T03687 C37GOB 90667455 IC50 = 37710 nM T03687 CJO6T1 91810840 IC50 = 5300 nM T03687 C34WIG 92045024 IC50 = 35000 nM T03687 C9OC0F 101882265 IC50 = 65800 nM T03687 CS2UL0 117829456 IC50 = 34 nM T03687 C7L4OT 117829461 IC50 = 120 nM T03687 C50VUN 117829462 IC50 = 41 nM T03687 CSU52M 118656852 IC50 = 500 nM T03687 CB6AJ9 118656853 IC50 = 200 nM T03687 C1JFZ7 118714371 IC50 = 55800 nM T03687 C2M5OR 118714376 IC50 = 18300 nM T03687 CY4GN9 118714377 IC50 = 47200 nM T03687 CI8G4X 118737400 IC50 = 10600 nM T03687 CL3M2F 121499152 IC50 > 33330 nM T03687 C28JVO 122192004 IC50 > 10000 nM T03687 CF2D8U 122192005 IC50 > 10000 nM T03687 C3V5ND 122550211 IC50 > 10000 nM T03687 CZE35C 122648343 IC50 > 1000 nM T03687 C54RNT 122648367 IC50 > 1000 nM T03687 C1UVI7 122648600 IC50 > 1000 nM T03687 CMX59K 122648648 IC50 > 1000 nM T03687 CVZ64I 122648649 IC50 > 1000 nM T03687 CV9I8D 127030313 IC50 = 8900 nM T03687 C6X3HG 132145728 IC50 = 1915 nM T03687 C8O9DP 132157820 IC50 = 1530 nM T03687 C4KE3N 132938351 IC50 > 10000 nM T03687 C05FVT 134492522 IC50 > 10000 nM T03687 C14FWK 135348858 IC50 = 38200 nM T03687 CDY18W 135407493 IC50 > 100000 nM T03687 CW2I4R 135412048 IC50 > 100000 nM T03687 C7U0AV 135412194 IC50 > 100000 nM T03687 CS54TL 135437514 IC50 > 100000 nM T03687 C36MUC 135441620 IC50 > 100000 nM T03687 CRB8M1 135444536 IC50 > 100000 nM T03687 CX5D6J 135446479 IC50 = 74100 nM T03687 C1TOK2 135449197 IC50 > 100000 nM T03687 CW25GL 135462117 IC50 > 100000 nM T03687 CCL28F 135473106 IC50 > 100000 nM T03687 CYA60G 135497781 IC50 > 100000 nM T03687 C8X5LO 135928012 Ki = 1400 nM T03687 CI2YE8 135928628 IC50 > 100000 nM T03687 C50NIS 136025837 IC50 > 100000 nM T03687 C4OS0V 136025842 IC50 > 100000 nM T03687 CX7Z5B 136025843 IC50 > 100000 nM T03687 CB8EM9 136025984 IC50 > 100000 nM T03687 C49MUG 136025986 IC50 > 100000 nM T03687 CH7Y3C 136086920 IC50 > 100000 nM T03687 C3VDL5 136086921 IC50 > 100000 nM T03687 C9GOB5 136086922 IC50 > 100000 nM T03687 CE3ZL7 136086923 IC50 > 100000 nM T03687 CJZ5F3 136086924 IC50 = 11700 nM T03687 CT19ND 136110961 IC50 > 100000 nM T03687 CY9U0E 136173089 IC50 > 50000 nM T03687 CRPN39 136645466 IC50 > 10000 nM T03687 C67EFJ 137628684 IC50 > 1000 nM T03687 CZ1FK2 137635119 IC50 > 50000 nM T03687 C5FHD3 137652442 IC50 = 70 nM T03687 CCR5B3 137654793 IC50 = 8500 nM T03687 C1SBN5 137654946 IC50 = 1680 nM T03687 C76OGQ 137656942 IC50 = 13000 nM T03687 CAQ62X 137701235 Ki > 10000 nM T03687 CN2UH1 139303146 IC50 > 20000 nM T03687 C7XI0V 141764754 IC50 = 441 nM T03687 CKBF56 142506033 IC50 > 100000 nM T03687 CGNQ74 142506189 IC50 = 3335 nM T03687 C1T3IQ 142506210 IC50 = 34850 nM T03687 CP5HF8 142506225 IC50 = 5349 nM T03687 CV3QO5 145951170 IC50 > 10000 nM T03687 CKG98W 145953085 IC50 > 30000 nM T03687 C9IV1C 145959866 IC50 > 10000 nM T03687 CK1XI0 145960971 IC50 > 10000 nM T03687 CP53JS 145977717 IC50 > 10000 nM T03687 CWD0A9 145983712 Ki > 10000 nM T03687 C56MWZ 145986208 Ki > 10000 nM T03687 C0YXS8 147254231 IC50 = 7782 nM T03687 CN71OS 149405396 IC50 > 100000 nM T03687 C8S3MF 150076000 IC50 > 300 nM T03687 C9FIY4 153534005 IC50 > 10000 nM T03687 CA1J3N 155517086 IC50 = 9100 nM T03687 CL72ME 155517175 IC50 > 10000 nM T03687 CY54TU 155518062 IC50 = 200 nM T03687 CEH2N5 155518106 IC50 > 100000 nM T03687 CAD06U 155519254 IC50 = 3070 nM T03687 CDY5H6 155519645 IC50 > 10000 nM T03687 CAZ3S7 155521187 IC50 > 30000 nM T03687 CZ75FW 155521272 IC50 = 15200 nM T03687 CIZ46A 155533876 IC50 = 8900 nM T03687 C6LB5D 155535084 IC50 = 25000 nM T03687 CTF98X 155537473 IC50 > 10000 nM T03687 CLD19W 155539311 IC50 > 10000 nM T03687 CS3GO2 155546558 IC50 = 9300 nM T03687 CGDF76 155554360 IC50 = 13000 nM T03687 CZDC03 155565491 IC50 > 30000 nM T03687 D00GBB 11449246 Ki = 55 nM T03687 D01YBR 44591988 IC50 = 13100 nM T03687 D02HVH 11427204 IC50 = 82 nM T03687 D02NWS 279980 IC50 = 430000 nM T03687 D03QOD 239512 IC50 = 510 nM T03687 D04KQF 6675804 Ki = 509.3 nM T03687 D05OVV 11993691 IC50 = 640 nM T03687 D09RKA 72946782 IC50 = 5000 nM T03687 D0E9DD 16095101 IC50 = 28000 nM T03687 D0K7QR 45269423 IC50 = 150 nM T03687 D0N9AK 44138031 IC50 = 12000 nM T03687 D0Q5DI 71462653 IC50 = 6720 nM T03687 D0R7JA 53344908 IC50 = 19.4 nM T03687 D0T0SK 44138032 IC50 = 2470 nM T03687 D0T4JQ 264 IC50 > 2000000 nM T03687 D0Z8PX 24757913 IC50 = 8330 nM T63298 D0E3TC 44259 IC50 = 83.5 nM T63298 CACS26 11561968 Ki > 2000 nM T63298 CU0E8O 11690457 Ki > 2000 nM T63298 CLS29B 46872626 IC50 > 10000 nM T63298 C1MR8Q 60097495 IC50 > 1000 nM T63298 CV63UL 67240318 IC50 > 10000 nM T63298 C2MD1Q 155513187 IC50 > 10000 nM T63298 D00ERW 44444843 Ki > 9570 nM T94479 D03ZBT 11626560 IC50 > 10000 nM T94479 D0EG1I 9926791 IC50 > 10000 nM T94479 D01NEC 51042438 IC50 = 60 nM T94479 D08UUL 46700756 IC50 = 382.18 nM T94479 D0CY1B 6420138 Ki = 540 nM T94479 D0E3TC 44259 IC50 = 0.553 nM T94479 D0VO5S 25118925 IC50 = 4 nM T94479 D0X2JM 56963011 IC50 = 2 nM T94479 D03BNU 59604787 IC50 > 3500 nM T94479 D0T3ME 156422 IC50 > 30000 nM T94479 CP9AM1 599038 Ki = 50 nM T94479 CE2G1Z 607858 Ki = 12 nM T94479 CY13FW 644243 IC50 = 950 nM T94479 CN8SU3 684961 Ki = 40 nM T94479 C5LHO7 753058 Ki = 540 nM T94479 C1SVD2 2132479 IC50 = 6000 nM T94479 CIOJ28 2422329 IC50 = 107 nM T94479 CNGT42 2959495 IC50 = 85 nM T94479 CS4P3Q 5000906 IC50 = 196 nM T94479 C6AD8F 5038004 Ki = 22 nM T94479 CDK3J0 5703619 IC50 = 0.75 nM T94479 CN6D5K 9801003 IC50 = 25000 nM T94479 C18HKQ 9885748 IC50 = 20000 nM T94479 CF9A5O 10125353 Ki = 69 nM T94479 CM79VS 10149184 Ki = 95 nM T94479 CC8XJ5 10171595 Ki = 110 nM T94479 CB28QI 10171783 Ki = 26 nM T94479 CL7FI4 10171832 Ki = 1900 nM T94479 CJ39UQ 10236371 Ki = 12 nM T94479 CM6DO0 11233873 IC50 = 2850 nM T94479 C0OZW2 11247002 IC50 = 560 nM T94479 CN16LZ 11269477 IC50 = 1550 nM T94479 COW1S8 11360518 IC50 = 1100 nM T94479 C9UI3O 11373846 IC50 = 1940 nM T94479 CONW29 11453116 IC50 = 4790 nM T94479 CS2YO1 11492918 Ki = 89 nM T94479 C4ARE5 11493905 IC50 = 9 nM T94479 C7HMO6 11526786 IC50 > 30000 nM T94479 C7IOJ0 11548023 IC50 = 1000 nM T94479 CO9KP5 11583459 IC50 > 10000 nM T94479 C71WAD 11615485 Ki = 340 nM T94479 CJS28X 11641672 IC50 = 2100 nM T94479 CM8W3K 11649421 IC50 > 20000 nM T94479 C65FVB 11694317 Ki = 1600 nM T94479 COH3C4 11697546 IC50 = 4500 nM T94479 C7DJS2 11713441 IC50 > 20000 nM T94479 CZY05V 11719421 IC50 = 2710 nM T94479 C5ISQ9 11751266 IC50 = 590 nM T94479 CHR92S 11858109 IC50 = 5700 nM T94479 CKV4G1 16079040 IC50 = 1400 nM T94479 CQK6C4 16099866 IC50 > 10000 nM T94479 CGC34R 16118737 IC50 > 100000 nM T94479 C54YXC 16121514 IC50 = 6.457 nM T94479 C9C5TV 17751819 IC50 = 120 nM T94479 CVS0T5 17754396 IC50 > 10000 nM T94479 C8AH1I 17758019 IC50 > 100000 nM T94479 C1GKL6 17758020 IC50 > 40000 nM T94479 CIE58R 17758239 IC50 = 18800 nM T94479 CO6LR5 17758240 IC50 > 40000 nM T94479 CWH37T 17758574 IC50 = 83100 nM T94479 C57NRL 17759787 IC50 > 40000 nM T94479 CG3VB6 23646578 IC50 = 70 nM T94479 C7YG1N 24759534 IC50 = 88 nM T94479 CQNP54 24764449 IC50 = 25000 nM T94479 C4Z9CN 24769780 IC50 = 65000 nM T94479 CJUK39 24770517 IC50 > 10000 nM T94479 C9PA0M 24807809 IC50 > 30000 nM T94479 C13QYB 24884503 IC50 > 2000 nM T94479 CL7V8R 25060409 IC50 = 97 nM T94479 CFU5E2 25060410 IC50 = 235 nM T94479 C3B8FI 25060411 IC50 = 76 nM T94479 C4CJX9 25060675 IC50 = 763 nM T94479 CRO09K 25211064 IC50 = 20000 nM T94479 CDR19S 25243801 IC50 = 9.1 nM T94479 C5Z3LI 44591740 IC50 > 30000 nM T94479 CVW08Q 44608012 IC50 = 107 nM T94479 C1SIK2 44620952 IC50 = 88 nM T94479 CDN3C4 44622839 Ki < 1 nM T94479 C5G0UA 44622840 Ki < 1 nM T94479 CQYO76 46192856 IC50 = 80 nM T94479 CU1Q0K 46192857 IC50 = 216 nM T94479 CQ82JV 46192858 IC50 = 72 nM T94479 CN0A1I 46192859 IC50 = 219 nM T94479 CM96WL 46192860 IC50 = 443 nM T94479 CDJS49 46192989 IC50 = 21 nM T94479 CS9T2M 46192991 IC50 = 93 nM T94479 CD4O0S 46192992 IC50 = 182 nM T94479 CPK5N7 46193129 IC50 = 77 nM T94479 CQ8YW5 46193130 IC50 = 254 nM T94479 C3VYA4 46193131 IC50 = 106 nM T94479 CS5Q2R 46193132 IC50 = 19 nM T94479 C52HOD 46193133 IC50 = 343 nM T94479 CZ58FY 46215814 IC50 = 6340 nM T94479 CY3HW5 46224684 IC50 > 10000 nM T94479 CLS29B 46872626 IC50 > 10000 nM T94479 CNTS27 46883044 Ki = 4 nM T94479 C0DB5Z 46883045 Ki = 13 nM T94479 C9WE4S 46883122 Ki = 800 nM T94479 CNTS75 46883123 Ki = 800 nM T94479 CJS68B 46883124 Ki = 31 nM T94479 CU3O2G 46883125 Ki = 550 nM T94479 CH9RV4 46883165 Ki = 39 nM T94479 CT1K6A 46883166 Ki = 410 nM T94479 CGZ1S4 46883167 Ki = 2200 nM T94479 C2VGJ9 46883168 Ki = 19 nM T94479 CT5V8K 46883169 Ki = 16 nM T94479 C60GAV 46929544 IC50 > 8000 nM T94479 CP34VL 46929748 IC50 > 1000 nM T94479 CJ2E9Q 46929857 IC50 > 25000 nM T94479 CI2T8K 51003535 IC50 = 521 nM T94479 CULS26 51003536 IC50 = 34 nM T94479 CL98KD 51003547 IC50 = 7000 nM T94479 CFQ5H6 51003548 IC50 = 10000 nM T94479 C8CGM9 51346966 IC50 = 399 nM T94479 CEQN27 52936621 Ki > 1000 nM T94479 CM24LF 52938983 IC50 < 1 nM T94479 CTUW53 53316599 IC50 > 20000 nM T94479 CEZ80N 53317553 IC50 = 29000 nM T94479 CP3S5T 53317852 IC50 = 379000 nM T94479 CWO65M 53317853 IC50 = 52000 nM T94479 COXV82 53317900 IC50 = 4000 nM T94479 C7I1JW 53319167 IC50 = 19000 nM T94479 C8X9HC 53319168 IC50 = 19000 nM T94479 C4RO9P 53319169 IC50 = 207000 nM T94479 C17ZLG 53320486 IC50 = 201000 nM T94479 CC30JO 53320487 IC50 = 191000 nM T94479 CWAT37 53320539 IC50 = 70000 nM T94479 C14HTQ 53320540 IC50 = 1900000 nM T94479 CU1PJ5 53321852 IC50 = 62000 nM T94479 CR1BI5 53321853 IC50 = 196000 nM T94479 CPO0X9 53323173 IC50 = 9000 nM T94479 CE6L3B 53323174 IC50 > 20000 nM T94479 C0Y1GX 53325333 IC50 = 223000 nM T94479 C6JA2K 53325839 IC50 > 20000 nM T94479 C8NA4L 53384644 IC50 = 20000 nM T94479 CM8JX1 56604907 IC50 = 1000 nM T94479 CT4E8R 56832546 IC50 = 12000 nM T94479 CQ57PE 57345536 IC50 = 2 nM T94479 C8R4FE 57991377 IC50 = 313.8 nM T94479 CT3EW2 59292007 IC50 > 1000 nM T94479 CXJ63M 59603829 IC50 = 110 nM T94479 CQEU96 59603842 IC50 = 8 nM T94479 CVRS14 59688971 IC50 = 2 nM T94479 C1MR8Q 60097495 IC50 > 2000 nM T94479 CUJ28O 67112053 IC50 = 1900 nM T94479 C2ZJC1 67113434 IC50 = 876 nM T94479 C83JZR 67160785 IC50 = 3 nM T94479 CZ3P5I 67160938 IC50 = 1 nM T94479 C5KOD3 67161433 IC50 = 37 nM T94479 CT04DK 67161469 IC50 = 1 nM T94479 CE5M9O 67161513 IC50 = 2 nM T94479 C5F8HT 67161588 IC50 = 11 nM T94479 C6K2VH 67161637 IC50 = 2 nM T94479 CG6XQ3 67161715 IC50 = 4 nM T94479 CP60OA 67161792 IC50 = 2 nM T94479 C52QDN 67161976 IC50 = 6 nM T94479 CRM5A3 67161981 IC50 > 2000 nM T94479 CWT8F6 67161992 IC50 = 6 nM T94479 C4XIR9 67162104 IC50 = 7 nM T94479 C9K3VX 67162133 IC50 = 16 nM T94479 C1YX5L 67162199 IC50 = 2 nM T94479 CNXU89 67162253 IC50 = 2 nM T94479 CSF3H9 67162282 IC50 = 6 nM T94479 CPB2W6 67162323 IC50 = 3 nM T94479 CE3GM8 67162496 IC50 = 29 nM T94479 CDH98A 67162510 IC50 = 5 nM T94479 C2G7FT 67162514 IC50 = 14 nM T94479 CIY82C 67162897 IC50 = 197 nM T94479 CU80DI 67162943 IC50 = 162 nM T94479 C1L2KG 67163351 IC50 = 13 nM T94479 CU2R1F 67163581 IC50 = 3 nM T94479 CV63UL 67240318 IC50 > 10000 nM T94479 C5DGR9 69036886 IC50 = 10000 nM T94479 C0M6FJ 70683203 IC50 > 2000 nM T94479 CD1ZJ8 70687431 IC50 = 3 nM T94479 C5D1LV 70687790 IC50 = 3311.31 nM T94479 C3C9NS 70689492 IC50 > 2000 nM T94479 CXSI14 71718330 IC50 > 100000 nM T94479 C1TM3P 71720141 IC50 > 100000 nM T94479 C0DL3F 72698602 IC50 < 1 nM T94479 CQ8ZU5 74538689 IC50 < 25 nM T94479 CU1AW9 76072947 IC50 = 501 nM T94479 CFY97V 76072948 IC50 < 25 nM T94479 CCP54M 76072949 IC50 = 25 nM T94479 C6F3UO 76072950 IC50 < 25 nM T94479 CT46PQ 76072951 IC50 < 25 nM T94479 CO3ML7 76072952 IC50 < 25 nM T94479 CJ13RN 76072989 IC50 < 25 nM T94479 CKSV46 76072990 IC50 = 25 nM T94479 CXEP31 76072991 IC50 < 25 nM T94479 C1O0RN 76073358 IC50 < 25 nM T94479 CV38TG 76073574 IC50 > 1000 nM T94479 CC26HG 76073575 IC50 < 25 nM T94479 CUWY13 76073576 IC50 > 1000 nM T94479 C6R3ME 76073577 IC50 = 501 nM T94479 CHO9D0 76073579 IC50 = 25 nM T94479 C1HW4B 89735655 IC50 = 1500 nM T94479 C8MIZ2 90194118 IC50 = 101 nM T94479 C2LAM7 126591927 IC50 = 23 nM T94479 CO47QJ 133054002 IC50 = 35 nM T94479 CU60YC 135431661 IC50 > 30000 nM T94479 CY4D8I 135566504 Ki = 773.4 nM T94479 CG3UZ1 135927974 Ki > 1000 nM T94479 CC73PA 138911338 IC50 = 8.9 nM T94479 C6VB3O 145925651 IC50 >= 5000 nM T94479 C8CIX0 145982744 IC50 > 1000 nM T94479 C03PYD 145986466 IC50 = 120 nM T94479 CSU93V 155077019 IC50 = 7.1 nM T94479 CL5DR0 155525783 IC50 = 7 nM T94479 CZQM57 155554194 IC50 = 625.68 nM T94479 D00ERW 44444843 Ki > 6668 nM T94479 D03MUZ 17759555 IC50 > 100000 nM T94479 D07OXC 11650194 IC50 = 10000 nM T94479 D09FFE 449241 IC50 = 80 nM T94479 D0I1FJ 11393719 IC50 = 270 nM T94479 D0L2WP 46225540 IC50 = 7 nM T94479 D0M5FF 5083 IC50 = 15 nM T80526 D09JEJ 24748573 IC50 = 11 nM T80526 D0E3TC 44259 IC50 = 844 nM T80526 D02GEJ 5326976 Ki = 112 nM T80526 CJH12X 537952 IC50 = 32200 nM T80526 CR9EJ0 11352337 Ki = 35 nM T80526 C8V7ZF 11352967 Ki = 37 nM T80526 CV78IN 16224258 IC50 = 190 nM T80526 CY8X0J 24811794 IC50 = 701 nM T80526 C4HY6I 44263430 Ki = 21 nM T80526 CYX19V 44263445 Ki = 78 nM T80526 C0RK5W 44263447 Ki = 62 nM T80526 CNZ19H 44263451 Ki = 342 nM T80526 C3VRO9 44557921 IC50 > 10000 nM T80526 CDK93W 56946894 IC50 < 3000 nM T80526 CE2DU7 56968171 Ki = 188 nM T80526 C4RIA1 56968172 Ki = 93 nM T80526 CYIO69 56968174 Ki = 31 nM T80526 CT1ZJ3 56968175 Ki = 55 nM T80526 C73NVJ 56968176 Ki = 44 nM T80526 C0MS9N 56968177 Ki = 83 nM T80526 C8WDK1 57342036 IC50 = 11 nM T80526 C0I6SZ 57342039 IC50 = 32000 nM T80526 CA7BS4 57342210 IC50 = 63 nM T80526 CVBF89 57342215 IC50 = 25000 nM T80526 C8P1ZB 57342375 IC50 = 5300 nM T80526 CH6RV3 57342376 IC50 = 3300 nM T80526 C65NOS 57342377 IC50 = 1700 nM T80526 C8TFC7 57342378 IC50 = 1200 nM T80526 CZ0R4K 57342379 IC50 = 5800 nM T80526 C8U4MB 57342380 IC50 = 1800 nM T80526 CJSO14 57342381 IC50 = 2800 nM T80526 CW3P9K 57342382 IC50 = 4300 nM T80526 CFX60S 57342541 IC50 = 1600 nM T80526 CF9BZ1 57342542 IC50 = 2900 nM T80526 C2C4XB 57342543 IC50 = 4300 nM T80526 C9XPF2 57342544 IC50 = 2700 nM T80526 C9MA4U 57342545 IC50 = 3000 nM T80526 CWZY51 57342546 IC50 = 8200 nM T80526 CK9IC1 57342547 IC50 = 3100 nM T80526 CO14NX 57342548 IC50 = 5700 nM T80526 CTNX36 57342718 IC50 = 2400 nM T80526 C8G6RK 57342719 IC50 = 2100 nM T80526 CJ9OF3 57400663 Ki = 24 nM T80526 CV63UL 67240318 IC50 > 10000 nM T80526 CDE3Y9 76321032 IC50 < 4000 nM T80526 C4T7YB 127025199 IC50 = 4.6 nM T80526 CP02TW 127025200 IC50 = 10 nM T80526 C57ECS 127025201 IC50 = 280 nM T80526 CP31UE 127025202 IC50 = 10 nM T80526 CHP6R9 127025499 IC50 = 12 nM T80526 CY37QE 127025500 IC50 = 12 nM T80526 CR59LY 127026094 IC50 = 11 nM T80526 CWIG59 127026095 IC50 = 9.8 nM T80526 C45BZG 127026096 IC50 = 160 nM T80526 C0HLT9 127026097 IC50 = 19 nM T80526 CW5JB1 127026098 IC50 = 14 nM T80526 CL4CG5 127026727 IC50 = 13 nM T80526 CO6X5B 127026728 IC50 = 11 nM T80526 CA5XG8 127026729 IC50 = 9.5 nM T80526 C6EIR3 127027657 IC50 = 9.6 nM T80526 C1MF5T 127029513 IC50 = 8.8 nM T80526 C86HPW 155518524 IC50 = 99000 nM T80526 D0CP3M 5149739 Ki = 270 nM T80526 D0K6BI 46943415 Ki = 21 nM T80526 D0US9O 45275255 IC50 = 2.7 nM T00099 D0G5ZE 72430 IC50 = 40 nM T00099 CXQL97 455769 IC50 = 25 nM T00099 CYW67U 455772 IC50 = 400 nM T00099 CC36MD 455773 IC50 = 140 nM T00099 CX8G9N 7299379 IC50 = 4.9 nM T00099 CI1Y6K 9822962 IC50 = 20 nM T00099 CYAC30 9910792 Ki = 7000 nM T00099 CV0CI4 10216098 IC50 = 35 nM T00099 CP8F0G 11157188 IC50 = 88.6 nM T00099 CFD37G 11157382 IC50 = 75.9 nM T00099 CI1WP6 11157406 IC50 = 38 nM T00099 CZ8L6J 11169393 IC50 = 222 nM T00099 C7T1AD 11180278 IC50 = 25 nM T00099 CK87ZO 11180469 IC50 = 48.7 nM T00099 CN0F8E 11199915 IC50 = 40 nM T00099 CMJX86 11203723 IC50 = 138 nM T00099 CGC7Z0 11203895 IC50 = 553.2 nM T00099 C0NJS1 11227053 IC50 = 105 nM T00099 C5HI9C 11273094 IC50 = 150.9 nM T00099 C5IO1M 11307066 IC50 = 8 nM T00099 CQJ4A5 11421890 IC50 = 150 nM T00099 C0JYZ9 11444285 IC50 = 85.5 nM T00099 C8B4LD 11444648 IC50 = 354.1 nM T00099 CV3D4Q 11467489 IC50 = 905 nM T00099 C20DLA 11489977 IC50 = 55.4 nM T00099 C3USR9 11543714 IC50 > 5000 nM T00099 C17OJS 11572844 IC50 > 5000 nM T00099 C6UAV3 11632008 IC50 > 5000 nM T00099 C91JNO 11639020 IC50 > 5000 nM T00099 C4MCW2 11646889 IC50 > 5000 nM T00099 CH20JE 11652994 IC50 > 5000 nM T00099 CKVL15 11852777 IC50 = 270 nM T00099 CUA19Y 16760339 Ki = 250 nM T00099 CG2OR8 18394274 IC50 = 30 nM T00099 C2GXK0 23240732 Ki = 4500 nM T00099 C52GAL 23240733 Ki = 1800 nM T00099 CT6PW7 23240734 Ki = 280 nM T00099 CJD86W 23240735 Ki = 680 nM T00099 C5SX7Z 23240736 Ki = 320 nM T00099 C6YW0C 23240737 Ki = 200 nM T00099 C15TFI 23240738 Ki = 200 nM T00099 C2NRA7 23240739 Ki = 52 nM T00099 C5UQT7 23240740 Ki = 8.5 nM T00099 CI89XA 23240741 Ki = 75 nM T00099 CAEG80 44343472 Ki < 4000 nM T00099 C1IPZ6 44343473 Ki = 1000 nM T00099 CN5GQ3 44343531 Ki = 15000 nM T00099 C15XLB 44343546 Ki = 320 nM T00099 CB53OZ 44343547 Ki = 1000 nM T00099 C63ZYT 44343548 Ki = 120 nM T00099 C02RUT 44343554 Ki = 3400 nM T00099 C60EVR 44343557 Ki = 320 nM T00099 C1WM7R 44343562 Ki = 160 nM T00099 CGN37W 44343594 Ki = 800 nM T00099 C47KQO 44343612 Ki = 200 nM T00099 C3V5XU 44343661 Ki = 100 nM T00099 CVR40J 44343678 Ki = 40000 nM T00099 C4G1DX 44343691 Ki = 69 nM T00099 C7LH3U 44343713 Ki = 1400 nM T00099 CQ6G9B 44343725 Ki = 76000 nM T00099 CU4DC6 44343744 Ki = 500 nM T00099 C8SFT5 44343749 Ki = 80 nM T00099 C7L2RA 44343763 Ki = 210 nM T00099 C0OSC3 44343848 Ki = 9500 nM T00099 CI1RC2 44343891 Ki = 2000 nM T00099 CNO65Y 44343910 Ki = 4000 nM T00099 C17NVX 44343911 Ki = 200 nM T00099 CVKL43 44343918 Ki = 96 nM T00099 CFR7P1 44343971 Ki = 20000 nM T00099 CIF9O3 44344001 Ki > 5000 nM T00099 CE7YB4 44344038 Ki = 5000 nM T00099 CSWU72 44344051 Ki = 1800 nM T00099 CUGS86 44351795 IC50 > 1000 nM T00099 C2QZ8I 44351809 IC50 = 500 nM T00099 CS35JT 44351836 IC50 = 100 nM T00099 C3W0QF 44351854 IC50 = 100 nM T00099 CAVC51 44351862 IC50 = 100 nM T00099 C8MCZ5 44351868 IC50 = 100 nM T00099 CGD4J3 44351869 IC50 = 55 nM T00099 CW0U7T 54243404 IC50 > 1000 nM T00099 C2Y6TO 73347008 Ki = 1800 nM T00099 CC2LB9 90663209 Ki = 1400 nM T00099 C4ZH1J 90663211 Ki = 33000 nM T00099 CQ42NT 90663212 Ki = 16000 nM T00099 C52LCE 90663213 Ki = 1300 nM T00099 D06FFP 443118 IC50 = 7000 nM T00099 D0V6DX 10640 IC50 > 5000 nM T25889 C8QM7B 6852376 EC50 = 71 nM T25889 C3BPW2 9938390 Ki = 29 nM T25889 CDW80I 10058098 EC50 = 5200 nM T25889 C3DQ2N 14182914 Ki = 4400000 nM T25889 C1L2KH 15120210 EC50 > 10000 nM T25889 COF34S 16100296 Ki = 254 nM T25889 CR06WQ 20742348 Ki = 110 nM T25889 CQUB12 44304524 Ki = 300 nM T25889 CSG47O 44304525 Ki > 2000 nM T25889 CJCT80 44304570 Ki > 2000 nM T25889 CVG1W6 44304581 Ki > 2000 nM T25889 C3ET1U 44304582 Ki > 2000 nM T25889 CCR41L 44304622 Ki = 33 nM T25889 CQ6Z2N 44304623 Ki > 2000 nM T25889 CM5EP0 44304770 Ki = 14 nM T25889 C2V6RG 44304771 Ki = 1000 nM T25889 C4D7PC 44304787 Ki > 2000 nM T25889 CMQY30 44304788 Ki = 317 nM T25889 CT5Z3Y 44304825 Ki = 144 nM T25889 C6ZB8E 44304828 Ki > 2000 nM T25889 CX3VC2 44304835 Ki = 20 nM T25889 C6UT0A 44304913 Ki > 2000 nM T25889 C1I0RU 44304965 Ki = 610 nM T25889 CTH50C 44304982 Ki > 2000 nM T25889 CLB1S3 44304993 Ki = 17 nM T25889 CJA5G3 73345411 Ki = 4.2 nM T25889 CHJ5Y9 73346936 Ki = 2.6 nM T25889 CKFB13 73351491 Ki = 3.9 nM T25889 CW12RO 90662881 Ki = 0.88 nM T25889 CC6VY4 90662882 Ki = 7.8 nM T25889 C6QWZ1 90662885 Ki = 1.7 nM T25889 CH21ZL 90662895 Ki = 1.9 nM T25889 C0MJ4E 90662897 Ki = 2.5 nM T25889 CL89JV 90662898 Ki = 1.7 nM T38763 D0D4YZ 45375808 EC50 = 34 nM T38763 D0NI0C 21704 IC50 = 50000 nM T38763 D04KJT 56640146 EC50 = 1.8 nM T38763 D09RVI 23649154 EC50 = 2.9 nM T38763 D09ZZW 503536 IC50 = 1500 nM T38763 D0H7QU 56934415 IC50 = 20 nM T38763 D05DDN 11561383 EC50 = 9 nM T38763 D0FY6Q 491098 IC50 = 1400 nM T38763 C3FDG1 10347 IC50 = 18000 nM T38763 CAU7R2 21919 IC50 > 50000 nM T38763 C2TXC4 69732 IC50 > 50000 nM T38763 C4Q7OV 100253 EC50 > 50000 nM T38763 CC90DA 102213 IC50 = 47000 nM T38763 CY8EA3 122619 EC50 = 1200 nM T38763 C3DNF6 129764 IC50 = 15200 nM T38763 CEDS79 308117 IC50 > 50000 nM T38763 CR5C8M 447368 IC50 = 1700 nM T38763 C6TL9M 447369 IC50 = 8600 nM T38763 CVWE08 490741 IC50 = 4000 nM T38763 CAJ64Q 490750 IC50 = 400 nM T38763 CE12XT 490759 IC50 = 400 nM T38763 C42YHR 490778 IC50 = 2000 nM T38763 C1UIA3 490946 IC50 = 12000 nM T38763 C16TPS 490947 IC50 = 3000 nM T38763 CPSU72 490960 IC50 = 2000 nM T38763 C6KXE5 490973 IC50 = 7000 nM T38763 CT2L0H 491062 IC50 = 19 nM T38763 CFR74W 491094 IC50 = 13000 nM T38763 C6NUQ8 491096 IC50 = 19000 nM T38763 CRKD18 491097 IC50 = 10000 nM T38763 C7PN8E 491099 IC50 = 8600 nM T38763 CD8H3K 491103 IC50 = 3400 nM T38763 CJO5W0 491105 IC50 > 30000 nM T38763 CZ4QO0 491107 IC50 = 13000 nM T38763 CQSC34 491108 IC50 = 3700 nM T38763 CC0EK2 491110 IC50 = 4600 nM T38763 CDU7L1 491113 IC50 = 1600 nM T38763 CMO49H 491114 IC50 = 4300 nM T38763 CK8YA4 491116 IC50 = 6330 nM T38763 CNY6P4 491117 IC50 = 1800 nM T38763 C5XH3V 491118 IC50 = 12000 nM T38763 C3DW0I 491125 IC50 = 1500 nM T38763 CMQ28J 491128 IC50 = 50 nM T38763 C2PY1G 491132 IC50 = 100 nM T38763 C38GLE 491135 IC50 = 700 nM T38763 C5FGU1 491140 IC50 = 20 nM T38763 C1DNW7 491141 IC50 = 37 nM T38763 CT7RW1 491142 IC50 = 460 nM T38763 CN5RI4 491145 IC50 = 90 nM T38763 CU14SH 491146 IC50 = 8 nM T38763 CKT67Q 491147 IC50 = 120 nM T38763 C6OL2A 491148 IC50 = 150 nM T38763 CANQ51 491166 IC50 = 140 nM T38763 C4SGH3 491215 IC50 = 400 nM T38763 CK0XS2 493225 EC50 > 50000 nM T38763 CEM6N5 493415 IC50 = 8000 nM T38763 CR67CJ 493416 IC50 = 11000 nM T38763 C84QRW 493418 IC50 = 5700 nM T38763 C8EDA0 500900 EC50 = 300 nM T38763 C4DFR3 500902 EC50 = 2800 nM T38763 C2BSI5 503516 IC50 = 14000 nM T38763 CFRT87 503517 IC50 = 5000 nM T38763 C37MIA 503526 IC50 = 1000 nM T38763 CT07LB 504674 IC50 = 5700 nM T38763 CVL47E 504675 IC50 = 8000 nM T38763 CT81MP 504676 IC50 = 3500 nM T38763 CO6JZ2 504677 IC50 = 9100 nM T38763 C56ABH 504678 IC50 = 53000 nM T38763 CZK2Q1 504679 IC50 = 8600 nM T38763 C9FI5K 504680 IC50 = 11000 nM T38763 C8IFN4 504681 IC50 = 15000 nM T38763 CTM24V 504682 IC50 = 8000 nM T38763 CCF82A 504683 IC50 = 1400 nM T38763 C9A2GM 504684 IC50 = 3200 nM T38763 C6F8LT 504685 IC50 = 1800 nM T38763 C9Q1YW 504687 IC50 = 800 nM T38763 C3UZA8 504688 IC50 = 6000 nM T38763 C58KRG 504689 IC50 = 8000 nM T38763 CLXA25 504690 IC50 = 2700 nM T38763 CZX4V6 504691 IC50 = 3100 nM T38763 CYR07P 504692 IC50 = 11000 nM T38763 CJ0Z2Q 504693 IC50 = 37 nM T38763 C4XGM1 510626 IC50 = 350 nM T38763 C7E1WM 510633 IC50 = 5000 nM T38763 C4QJ1R 510646 IC50 = 44000 nM T38763 CI05HV 510665 IC50 = 16700 nM T38763 CQU18K 510674 IC50 = 3900 nM T38763 CN94PC 510692 IC50 = 10000 nM T38763 CMU9Q8 510698 IC50 = 25000 nM T38763 CF61MP 510705 IC50 = 16000 nM T38763 C9F0DP 510745 IC50 = 30000 nM T38763 CZ17SK 510792 IC50 = 47000 nM T38763 CTO28H 510839 IC50 > 50000 nM T38763 CMVB42 510844 IC50 = 4500 nM T38763 CO6VA0 510862 IC50 > 50000 nM T38763 CUWP10 510864 IC50 > 50000 nM T38763 CJ56OH 513150 IC50 < 6 nM T38763 CV9P7J 513870 EC50 = 7000 nM T38763 C5BN4U 513891 IC50 = 12000 nM T38763 CML9N5 513892 IC50 = 28000 nM T38763 CML6K9 513894 IC50 = 27000 nM T38763 CCS58A 513895 IC50 > 500000 nM T38763 CYH83S 513896 IC50 = 49000 nM T38763 CQO7W8 513897 IC50 = 76000 nM T38763 CN6LS1 513898 IC50 = 139000 nM T38763 CBJ1S6 513899 IC50 = 408000 nM T38763 CL3IJ7 513902 IC50 = 360000 nM T38763 C2IM7P 513903 IC50 = 186000 nM T38763 C4LR9N 513904 IC50 = 120000 nM T38763 C5GT1K 513905 IC50 = 58000 nM T38763 CVN79D 513906 IC50 = 20000 nM T38763 CGF30K 513907 IC50 = 62000 nM T38763 CEUG62 513908 IC50 = 44000 nM T38763 C60TID 513909 IC50 = 28000 nM T38763 C1IEQ4 513910 IC50 = 17000 nM T38763 CJ50YO 513911 IC50 = 5900 nM T38763 C05IUS 514257 EC50 = 6 nM T38763 C9VCM0 514258 IC50 = 30 nM T38763 CK8M6O 514262 IC50 = 90 nM T38763 CCRW58 514263 IC50 = 16 nM T38763 C6QRH4 514266 IC50 = 25 nM T38763 CC4U2P 514267 IC50 = 21 nM T38763 C1WOF8 514283 IC50 = 78 nM T38763 CJL15Q 514285 IC50 = 230 nM T38763 CBUX58 514293 IC50 = 80 nM T38763 CPI21K 516696 IC50 > 50000 nM T38763 C19CYX 516697 IC50 > 50000 nM T38763 CC1M3U 516699 IC50 > 50000 nM T38763 COT23S 516700 IC50 > 50000 nM T38763 CW2J4E 657131 IC50 = 100 nM T38763 CDU5A3 794768 IC50 = 619.44 nM T38763 CFU5G1 1269456 IC50 > 30000 nM T38763 CKI6L5 1269458 IC50 > 30000 nM T38763 C1QZP4 1286262 IC50 = 22000 nM T38763 CH37FY 1287042 IC50 = 1000 nM T38763 CDAV54 1308950 IC50 = 209.89 nM T38763 CSE3D0 1311270 IC50 = 990 nM T38763 C6V2UF 1317938 IC50 = 489.78 nM T38763 CL23YA 1379464 IC50 > 30000 nM T38763 CQC0A3 1379483 IC50 = 16000 nM T38763 C8Y0MZ 1379521 IC50 = 30000 nM T38763 CC6GS7 1380234 IC50 > 30000 nM T38763 CC5GE1 1384783 IC50 = 199.99 nM T38763 C2IHT3 1417800 IC50 = 5000 nM T38763 C07SDJ 1552027 IC50 = 1500 nM T38763 CS7H5N 1552029 IC50 = 700 nM T38763 C4GBI9 1565789 IC50 > 30000 nM T38763 C8KV9E 1583408 IC50 = 100 nM T38763 CC3K4L 1605277 IC50 = 750 nM T38763 CJT59B 1712167 IC50 > 30000 nM T38763 CGJ1P4 1722407 IC50 = 30000 nM T38763 CI04RH 1842471 IC50 = 539.51 nM T38763 CS7J6Z 1866916 IC50 = 1000 nM T38763 CE45QO 1886260 IC50 = 119.95 nM T38763 C7EFB1 1887699 IC50 = 1820 nM T38763 C8X5GB 1934431 IC50 > 30000 nM T38763 CW74JD 1958080 IC50 = 1000 nM T38763 C56DQB 1998838 IC50 = 200 nM T38763 C71MLS 2029569 IC50 = 15000 nM T38763 C4H2UC 2986648 IC50 = 4800 nM T38763 CC3A2G 3009857 EC50 > 50000 nM T38763 CV1OD2 3009858 EC50 > 50000 nM T38763 CK7ZG5 3009859 EC50 > 50000 nM T38763 CI2BN5 3009860 EC50 > 50000 nM T38763 C48ZYW 3009862 EC50 > 50000 nM T38763 CA7C6L 3009863 IC50 = 46000 nM T38763 CGWH27 3010939 IC50 > 100000 nM T38763 CI45RF 3010940 IC50 = 2250 nM T38763 CH8FY1 3010941 IC50 = 4000 nM T38763 CVHU24 3010942 IC50 > 100000 nM T38763 CTN40Q 3010943 IC50 = 51000 nM T38763 CUS35T 3010944 IC50 = 24000 nM T38763 C1VU5M 3010945 IC50 > 100000 nM T38763 C1HU3G 3010946 IC50 = 16200 nM T38763 C8TBM4 3010949 IC50 = 19000 nM T38763 CK65EZ 3012618 IC50 = 14000 nM T38763 C3E1ZI 3012981 IC50 = 5000 nM T38763 C2JEZ8 3012982 IC50 = 1400 nM T38763 CIFC56 3012983 IC50 = 11300 nM T38763 CUOH19 3012984 IC50 > 26000 nM T38763 C1TH6G 3012985 IC50 > 20000 nM T38763 CF2WT7 3012986 IC50 = 3100 nM T38763 CBW9R6 3012987 IC50 = 4900 nM T38763 CB64CG 3012988 IC50 = 2900 nM T38763 CZAH16 3012989 IC50 = 3300 nM T38763 C8VU7R 3012990 IC50 = 7700 nM T38763 C5SR3B 3012991 IC50 = 6400 nM T38763 CXS5D1 3012992 IC50 > 10000 nM T38763 CD0N5X 3012993 IC50 = 5100 nM T38763 CU5Q3V 3012994 IC50 = 2000 nM T38763 C7FNO8 3012995 IC50 = 900 nM T38763 CIX6K4 3013039 IC50 = 50000 nM T38763 CZP8B0 3013041 IC50 = 49000 nM T38763 CZE9V6 3535870 IC50 = 4000 nM T38763 C3EY6C 4369513 IC50 = 70 nM T38763 C83MIG 4369534 EC50 = 0.8 nM T38763 CMT3B2 5273318 IC50 > 50000 nM T38763 CLPG25 5273397 IC50 = 16000 nM T38763 CP4KF2 5273398 IC50 = 6000 nM T38763 C4Z0UW 5273399 IC50 > 100000 nM T38763 CM3PQ9 5273400 IC50 = 87000 nM T38763 CJI40L 5273401 IC50 > 100000 nM T38763 CBU5G3 5273402 IC50 = 29000 nM T38763 CHBO80 5273403 IC50 > 100000 nM T38763 CL87QY 5273404 IC50 > 100000 nM T38763 C7MJ0F 5273417 IC50 = 2900 nM T38763 C2JVW1 5273418 IC50 = 1500 nM T38763 C5SC2M 5273419 IC50 > 100000 nM T38763 CP2I1Q 5273420 IC50 = 73000 nM T38763 CV8OE1 5273421 IC50 = 68000 nM T38763 C8JDX6 5273422 IC50 = 3200 nM T38763 CC9SU8 5273423 IC50 = 9600 nM T38763 C9CY0L 5273424 IC50 = 26000 nM T38763 CT4QW6 5273425 IC50 = 21000 nM T38763 CGJ46F 5273426 IC50 = 10000 nM T38763 CL28NQ 5273427 IC50 = 2100 nM T38763 C4GSZ6 5273428 IC50 = 1300 nM T38763 C6UO5A 5273430 IC50 = 2900 nM T38763 CWC58H 5273431 IC50 = 13000 nM T38763 CM95OL 5273432 IC50 = 80000 nM T38763 CY19RZ 5273713 IC50 = 7000 nM T38763 C8VIP0 5273714 IC50 > 50000 nM T38763 CUR7W1 5273715 IC50 > 50000 nM T38763 CSIY93 5273716 IC50 = 13000 nM T38763 C1S7FX 5273717 IC50 > 50000 nM T38763 C5EI7A 5273719 IC50 = 6100 nM T38763 CXE2Y5 5273720 IC50 = 5000 nM T38763 C25PGY 5273721 IC50 = 3400 nM T38763 CSCH76 5273723 IC50 = 10000 nM T38763 C4LM1D 5273724 IC50 > 50000 nM T38763 CVA09O 5273725 IC50 > 50000 nM T38763 CK29LJ 5273728 IC50 = 5400 nM T38763 CMRQ48 5273729 IC50 = 2800 nM T38763 C23GCM 5273731 IC50 = 4400 nM T38763 C24VRZ 5273732 IC50 = 2800 nM T38763 C24NJY 5273733 IC50 = 4400 nM T38763 C3MQU6 5273734 IC50 = 3100 nM T38763 CK0S5X 5273735 IC50 = 8500 nM T38763 CCO3N5 5273736 IC50 = 2600 nM T38763 C8MQA3 5273737 IC50 = 3500 nM T38763 CKQW48 5273738 IC50 = 5200 nM T38763 CWL78I 5273739 IC50 = 6500 nM T38763 CO34QH 5273740 IC50 = 15000 nM T38763 C2TMC6 5273741 IC50 = 7000 nM T38763 C80NAU 5273742 IC50 = 1400 nM T38763 CBU4T0 5273743 IC50 = 5100 nM T38763 C1F8TX 5273744 IC50 = 4000 nM T38763 CQRH12 5273745 IC50 = 3900 nM T38763 C85DNB 5273746 IC50 = 6500 nM T38763 CE03XR 5273747 IC50 = 8500 nM T38763 CV86JC 5273748 IC50 = 3200 nM T38763 C7Q9BN 5273765 IC50 = 570 nM T38763 C72BQF 5275416 IC50 = 1900 nM T38763 CPKA37 5275418 IC50 = 3300 nM T38763 C64APQ 5275419 IC50 > 20000 nM T38763 C32ROZ 5275420 IC50 > 20000 nM T38763 CX8Y3M 5275421 IC50 > 20000 nM T38763 C0D6GM 5275422 IC50 = 190 nM T38763 C3F0XD 5275423 IC50 = 900 nM T38763 CWSM65 5275424 IC50 = 5100 nM T38763 CC3TQ4 5275425 IC50 = 1000 nM T38763 CEKM72 5275427 IC50 = 800 nM T38763 CB3VI4 5275428 IC50 = 700 nM T38763 C9C0SX 5275429 IC50 = 500 nM T38763 CB5DN3 5275430 IC50 = 11400 nM T38763 C7RVJ9 5275431 IC50 = 1700 nM T38763 C4DP3U 5275432 IC50 = 3200 nM T38763 CG5QM9 5275433 IC50 = 600 nM T38763 CKR1S8 5275434 IC50 > 20000 nM T38763 C9YCI1 5275435 IC50 = 600 nM T38763 CAYX59 5275436 IC50 > 20000 nM T38763 C5B2KX 5275437 IC50 = 700 nM T38763 CMBC61 5275438 IC50 > 20000 nM T38763 C6GS9M 5275439 EC50 = 6.7 nM T38763 CWD08Y 5275440 EC50 = 14.2 nM T38763 CMS5P6 5275441 EC50 > 50 nM T38763 C6SU7P 5275442 IC50 = 45 nM T38763 C58KCN 5275443 EC50 = 4.6 nM T38763 CLF2I9 5275444 EC50 = 1.5 nM T38763 C5YJN1 5275445 IC50 = 372 nM T38763 C48DRJ 5275446 EC50 = 4.5 nM T38763 CI2N5T 5275447 EC50 = 0.9 nM T38763 C3XUJ8 5275448 EC50 = 0.6 nM T38763 C2CZ6P 5275449 EC50 = 0.5 nM T38763 CXU6L9 5275450 EC50 = 0.5 nM T38763 CO17RX 5275451 EC50 = 2.6 nM T38763 CBF69J 5275452 IC50 = 11 nM T38763 C59ODA 5279449 IC50 = 80 nM T38763 CDXQ35 5279450 IC50 = 90 nM T38763 CAI02E 5279451 IC50 = 110 nM T38763 C7SF2A 5279452 IC50 = 120 nM T38763 CU9RN5 5279453 IC50 = 180 nM T38763 CB71TK 5279454 IC50 = 230 nM T38763 CQ0E1S 5279455 IC50 = 230 nM T38763 CO6L0Y 5279456 IC50 = 250 nM T38763 C45SCB 5279457 IC50 = 820 nM T38763 CKO37V 5279458 IC50 = 940 nM T38763 C6I8KZ 5279459 IC50 = 1000 nM T38763 C1DV5E 5279460 IC50 = 1000 nM T38763 C5S3BE 5279461 IC50 = 2200 nM T38763 C2H7VQ 5279462 IC50 = 370 nM T38763 CD6G7Y 5279463 IC50 = 500 nM T38763 CG0L1D 5279464 IC50 = 600 nM T38763 CB40UH 5279465 IC50 = 2600 nM T38763 C5TO7D 5279467 IC50 = 7000 nM T38763 CPW79T 5279468 IC50 = 6000 nM T38763 CZ52JX 5279469 IC50 = 6300 nM T38763 CW1JL6 5279470 IC50 = 7100 nM T38763 CE4V6R 5279471 IC50 = 15000 nM T38763 CBO28Z 5279472 IC50 = 14000 nM T38763 C3WQ7S 5279473 IC50 = 500 nM T38763 CI1D9T 5279474 IC50 = 1000 nM T38763 CI09FW 5279475 IC50 = 800 nM T38763 CYP6H4 5279476 IC50 = 2700 nM T38763 CR5GW3 5279477 IC50 = 60 nM T38763 C0T4NQ 5279478 IC50 > 100000 nM T38763 CIRP20 5279479 IC50 > 100000 nM T38763 C7OJ3T 5279480 IC50 = 12000 nM T38763 C23UWE 5279481 IC50 = 1900 nM T38763 CD7XJ5 5279482 IC50 = 15000 nM T38763 CW46CH 5279483 IC50 = 400 nM T38763 CWYU91 5742696 IC50 = 93000 nM T38763 CS3Z8I 5749224 IC50 > 30000 nM T38763 CO6M1D 5845808 IC50 = 250 nM T38763 C86TKB 6064166 IC50 = 7000 nM T38763 CNB2J8 6096788 IC50 > 50000 nM T38763 CUS7A1 6123445 IC50 = 580 nM T38763 C3VBL4 6264224 IC50 > 30000 nM T38763 CQ20AB 6479231 IC50 = 28000 nM T38763 CUAD01 6479232 IC50 = 16000 nM T38763 C5EUN9 6480674 IC50 = 6700 nM T38763 C5PH2N 6480675 IC50 = 1500 nM T38763 CYPN67 6480676 IC50 = 660 nM T38763 CJ4A1D 6480677 IC50 = 1300 nM T38763 CW85ZX 6480678 IC50 = 1400 nM T38763 CK95RD 6480679 IC50 = 3000 nM T38763 CB7HP8 6480680 IC50 = 2600 nM T38763 C4K3YA 6480681 IC50 = 3100 nM T38763 CZQJ81 6480682 IC50 = 3900 nM T38763 C5U0KX 6480683 IC50 = 4000 nM T38763 CYBV37 6480684 IC50 = 4600 nM T38763 C06UWY 6480685 IC50 = 5600 nM T38763 CFK8D9 6480686 IC50 = 6000 nM T38763 C0MON8 6480687 IC50 = 6900 nM T38763 C7LRC8 6480688 IC50 = 8700 nM T38763 CQB1A0 6480689 IC50 = 12000 nM T38763 C9UG1H 6480690 IC50 = 13000 nM T38763 CH6V1B 6480691 IC50 = 20000 nM T38763 CX3SC0 6480692 IC50 = 20000 nM T38763 C6G4TA 6480693 IC50 = 22000 nM T38763 CJO7W4 6480694 IC50 = 25000 nM T38763 C3MDK2 6480695 IC50 = 27000 nM T38763 C3IBA5 6480696 IC50 = 66000 nM T38763 C6Q1SD 6480697 IC50 > 100000 nM T38763 CF9N2Y 6480698 IC50 > 100000 nM T38763 CJ0V5N 6480699 IC50 > 100000 nM T38763 CTV6H8 6480700 IC50 > 100000 nM T38763 C27YZR 6480701 IC50 > 100000 nM T38763 CU51NM 6480702 IC50 = 200 nM T38763 CINM75 6480703 IC50 = 1300 nM T38763 CIE92V 6480704 IC50 = 11000 nM T38763 C25HVJ 6480705 IC50 > 100000 nM T38763 CAB75S 6480706 IC50 = 40 nM T38763 CDQ25X 6480707 IC50 = 580 nM T38763 C4UWZ7 6480708 IC50 = 1300 nM T38763 CKJ08I 6480709 IC50 = 1800 nM T38763 CI2YQ0 6480710 IC50 = 6900 nM T38763 C3XSM4 6480711 IC50 = 9400 nM T38763 C82TOU 6480712 IC50 = 15000 nM T38763 C21HJG 6480713 IC50 = 17000 nM T38763 CCJ18E 6480714 IC50 = 28000 nM T38763 CFXQ64 6480715 IC50 = 48000 nM T38763 C91QBI 6480716 IC50 = 44000 nM T38763 C01SGY 6480717 IC50 = 47000 nM T38763 C2L4ZG 6480718 IC50 = 73000 nM T38763 CEWU47 6480719 IC50 > 100000 nM T38763 CMFJ52 6480720 IC50 = 30 nM T38763 CIF0R5 6480721 IC50 = 70 nM T38763 C18NYQ 6480722 IC50 = 200 nM T38763 CR4FX2 6480723 IC50 = 310 nM T38763 C53YGX 6480724 IC50 = 5500 nM T38763 CH62BJ 6480885 IC50 = 62 nM T38763 C13HGI 6480886 IC50 = 63 nM T38763 C4S2PR 6480887 IC50 = 98 nM T38763 C6H4YC 6480888 IC50 = 43 nM T38763 C8GXD7 6480889 IC50 = 19 nM T38763 CC2ZG5 6480891 IC50 = 39 nM T38763 C1IYA4 6480892 IC50 = 18 nM T38763 CMBR61 6480893 IC50 = 11 nM T38763 CNEV49 6480894 IC50 = 8 nM T38763 CJ04UM 6480895 IC50 = 17 nM T38763 C0SI7D 6480896 IC50 = 11 nM T38763 C3CAN6 6480897 IC50 = 7 nM T38763 CJL3M1 6480899 IC50 = 12 nM T38763 CQ8TX5 6480900 IC50 = 12 nM T38763 CZ6UD3 6480907 IC50 = 448 nM T38763 C8PJW6 6480915 IC50 = 68 nM T38763 CT3UR7 6480916 IC50 = 47 nM T38763 CHZ60K 6480918 IC50 = 283 nM T38763 C1DE3X 6480919 IC50 = 72 nM T38763 CU49LS 6480920 IC50 = 49 nM T38763 C9PV0O 6480921 IC50 = 18 nM T38763 CP21VD 6480922 IC50 = 228 nM T38763 CPI9Z0 6480923 IC50 = 920 nM T38763 CZP64J 6480924 IC50 = 147 nM T38763 C3NZ7O 6480925 IC50 = 78 nM T38763 CRK90Z 6480926 IC50 = 78 nM T38763 CXUF67 6480927 IC50 = 18 nM T38763 CLW2H4 6480928 IC50 = 332 nM T38763 CYT19Q 6480929 IC50 = 134 nM T38763 C19MLS 6480930 IC50 = 69 nM T38763 C42EOG 6480931 IC50 = 31 nM T38763 CGM32K 6480932 IC50 = 9 nM T38763 C4UTI6 6480933 IC50 = 9 nM T38763 CS96GD 6480934 IC50 = 9 nM T38763 CC38KX 6480935 IC50 = 9 nM T38763 CR4MT9 6480936 IC50 = 9 nM T38763 C21OEX 6483672 IC50 = 5200 nM T38763 CVU36F 6559079 IC50 > 20000 nM T38763 C6OF2J 6914644 IC50 = 3100 nM T38763 CK5N3Q 9862510 IC50 = 890 nM T38763 CWF08N 9901786 IC50 = 51 nM T38763 C3KD2P 9912708 IC50 = 700 nM T38763 CJ3O6C 9946979 IC50 = 25000 nM T38763 CS7F4Y 9971466 IC50 > 50000 nM T38763 CC2M7V 10097021 EC50 = 100 nM T38763 C70KEC 10116001 IC50 = 1500 nM T38763 C1JN2O 10120254 IC50 = 300 nM T38763 C6W9EP 10122014 IC50 = 18 nM T38763 CGH72Q 10137290 IC50 = 1600 nM T38763 CA5VJ1 10137405 IC50 = 15000 nM T38763 C8JV9F 10140778 IC50 = 1000 nM T38763 CU1JZ6 10141859 IC50 = 300 nM T38763 C64RQF 10143976 IC50 = 98 nM T38763 C7SO4T 10144617 IC50 = 2400 nM T38763 CZRS52 10144618 IC50 = 480 nM T38763 CC17AG 10158598 IC50 = 3200 nM T38763 C53JUD 10160567 IC50 = 2100 nM T38763 CWS2N1 10163324 IC50 = 580 nM T38763 C4A0HE 10184305 IC50 = 1800 nM T38763 CWP01B 10184365 IC50 = 1700 nM T38763 C3B2KX 10185481 IC50 = 1300 nM T38763 C6BHR9 10187091 IC50 = 290 nM T38763 CWM73X 10188077 IC50 = 100 nM T38763 CUK70S 10188179 IC50 = 50 nM T38763 C9NSJ0 10188772 IC50 = 22 nM T38763 CLY58V 10204044 IC50 = 1600 nM T38763 CDQ6H2 10209030 EC50 = 2200 nM T38763 C7A6HW 10226237 IC50 = 6700 nM T38763 C1FN2L 10229600 IC50 = 980 nM T38763 C2SR8N 10229601 IC50 = 340 nM T38763 C58FZS 10230222 EC50 = 3700 nM T38763 C5AXK6 10230544 IC50 = 760 nM T38763 CXI45Z 10231235 IC50 = 170 nM T38763 CUQP17 10275464 IC50 = 2300 nM T38763 CF13ZR 10275979 IC50 = 800 nM T38763 CKYP72 10292795 IC50 = 4000 nM T38763 C8SAX3 10297424 IC50 = 1200 nM T38763 CJ49FU 10298006 IC50 = 1200 nM T38763 C3W1VG 10299516 IC50 = 1300 nM T38763 C7RZP3 10303157 IC50 = 41 nM T38763 C4PKG8 10339613 IC50 = 4000 nM T38763 C78QUL 10471727 IC50 = 1800 nM T38763 CPZN90 11163587 IC50 = 25 nM T38763 CN32QM 11163833 EC50 = 3200 nM T38763 CRQ4A5 11177350 IC50 = 230 nM T38763 CH9K7T 11209864 IC50 = 340 nM T38763 CVT5R3 11235044 IC50 = 120 nM T38763 C6H0AX 11301804 IC50 = 120 nM T38763 CFM64B 11350255 IC50 = 2200 nM T38763 C7PTY5 11370785 IC50 = 66 nM T38763 CU24SI 11418422 IC50 = 58 nM T38763 CW4IG6 11453453 IC50 = 120 nM T38763 CBRV21 11484451 IC50 = 4.8 nM T38763 CPJC40 11488676 IC50 = 41 nM T38763 C6L5VS 11492747 IC50 > 20000 nM T38763 CN60AC 11493106 IC50 = 4600 nM T38763 CZ3R5K 11493372 IC50 = 2000 nM T38763 C1P9CJ 11500555 IC50 = 1200 nM T38763 C8GX0M 11509370 IC50 = 25000 nM T38763 CS6WR0 11515367 IC50 = 1900 nM T38763 CEI0P1 11517044 IC50 = 5000 nM T38763 CFEQ18 11522600 IC50 = 5950 nM T38763 C9AJ7K 11522754 IC50 = 170 nM T38763 CS8IK0 11525611 IC50 = 17 nM T38763 CW1T5G 11529046 IC50 = 7000 nM T38763 CD15EY 11536839 IC50 = 30000 nM T38763 COT4A5 11538841 IC50 = 9940 nM T38763 CN0YM6 11543734 IC50 = 4700 nM T38763 C7IHE5 11553664 IC50 = 3000 nM T38763 CJUW59 11554181 IC50 = 27000 nM T38763 C2XS1F 11570085 IC50 = 200 nM T38763 C4GIZ2 11572713 IC50 = 11000 nM T38763 C8N7OZ 11580282 IC50 = 1800 nM T38763 CDL32W 11580625 IC50 = 2100 nM T38763 CADP43 11581550 IC50 = 750 nM T38763 CDB9S2 11582187 IC50 = 8000 nM T38763 C7I6XM 11582786 IC50 = 1900 nM T38763 CNU24V 11587498 IC50 = 5400 nM T38763 CGI91Y 11587905 IC50 = 17200 nM T38763 C3V5WI 11588555 IC50 > 20000 nM T38763 CVWE70 11595036 IC50 = 13800 nM T38763 C1Q6YC 11596698 IC50 > 10000 nM T38763 CC0R4K 11601725 IC50 > 20000 nM T38763 C3XQ8Y 11602097 IC50 = 1500 nM T38763 CNBS60 11602287 IC50 = 3200 nM T38763 C5R9DZ 11602933 IC50 = 77 nM T38763 C8UZ7Y 11604214 IC50 > 20000 nM T38763 CX7SL6 11604364 IC50 = 1000 nM T38763 CD4QY7 11604714 IC50 = 200 nM T38763 C7Z8YV 11606349 IC50 = 100 nM T38763 CJ6A1E 11611706 IC50 = 200 nM T38763 C8R2ZQ 11616882 IC50 = 2850 nM T38763 CO0WI4 11617192 IC50 = 130 nM T38763 CK43ND 11617889 IC50 = 2000 nM T38763 CX4I9C 11624253 IC50 = 770 nM T38763 CL1D3X 11624656 IC50 = 140 nM T38763 C5F9KG 11625951 IC50 = 2000 nM T38763 C2KR4Y 11626440 IC50 = 1000 nM T38763 CPE64V 11631291 IC50 = 320 nM T38763 CET3I2 11631314 IC50 = 17600 nM T38763 C8I2EW 11631571 IC50 = 1900 nM T38763 C6C0RS 11631847 IC50 = 5800 nM T38763 CI57WD 11632629 IC50 > 10000 nM T38763 CS4PA7 11640450 IC50 = 700 nM T38763 C9YOQ6 11645113 IC50 = 10000 nM T38763 CASG93 11645283 IC50 = 550 nM T38763 C79LIJ 11645475 IC50 > 20000 nM T38763 C78WSD 11654506 IC50 = 1700 nM T38763 C5WK1T 11660780 IC50 = 80 nM T38763 CQP07A 11661726 IC50 = 15000 nM T38763 C94BND 11668743 IC50 = 3000 nM T38763 C92KUO 11669161 IC50 = 1000 nM T38763 CXN9B2 11675585 IC50 = 6500 nM T38763 CI4HD8 11675604 IC50 > 10000 nM T38763 C8SGU5 11680778 IC50 = 14500 nM T38763 CAWZ70 11682794 IC50 = 900 nM T38763 CIYW64 11686018 IC50 = 61 nM T38763 CG49LT 11687835 IC50 = 8100 nM T38763 C3CZ9E 11689664 IC50 = 10000 nM T38763 CS1VP4 11690668 IC50 = 90 nM T38763 C71QVJ 11695055 IC50 = 15000 nM T38763 CM2X4B 11695645 IC50 = 210 nM T38763 CZG2V6 11709554 IC50 = 2300 nM T38763 CC9JR3 11710702 IC50 = 190 nM T38763 C2B9UH 11712094 IC50 = 200 nM T38763 CZV53X 11716351 IC50 = 6300 nM T38763 CK4XG6 11717072 IC50 > 33000 nM T38763 CDY1W4 11717209 IC50 = 5360 nM T38763 C67VRU 11717942 IC50 = 260 nM T38763 CX1D4O 11779681 IC50 = 8200 nM T38763 C36JAO 11844936 IC50 = 23 nM T38763 CS57HG 11844937 IC50 = 18 nM T38763 CH5M6Z 11844938 IC50 = 63 nM T38763 CNTQ57 11844939 IC50 = 24 nM T38763 C1KIF8 11845100 IC50 = 13 nM T38763 CP3L9V 11845101 IC50 = 15 nM T38763 C89VSG 11845102 IC50 = 29 nM T38763 C6O3FT 11845103 IC50 = 32 nM T38763 CMC26U 11845261 IC50 = 580 nM T38763 CY32GI 11845262 IC50 = 90 nM T38763 CHJ56S 11845263 IC50 = 188 nM T38763 CI19TD 11845264 IC50 = 53 nM T38763 C67YRX 11845265 IC50 = 150 nM T38763 C57TSE 11845266 IC50 = 100 nM T38763 CAYC38 11845432 IC50 = 350 nM T38763 CURV40 11845433 IC50 = 1100 nM T38763 COH3U5 11845434 IC50 = 930 nM T38763 CQ0ZR8 11845435 IC50 = 380 nM T38763 C2NY6G 11845436 IC50 = 12 nM T38763 C80YES 11845616 IC50 = 21 nM T38763 C0HTL3 11845617 IC50 = 13 nM T38763 CWLS20 11845618 IC50 = 21 nM T38763 C4JS8N 11845619 IC50 = 12 nM T38763 C2CWR5 11845798 IC50 = 18 nM T38763 CH5DT7 11845799 IC50 = 14 nM T38763 CJP09V 11845800 IC50 = 14 nM T38763 CQ2KX5 11845801 IC50 = 16 nM T38763 CF47CU 11845802 IC50 = 19 nM T38763 C5CHV6 11845985 IC50 = 32 nM T38763 C87QXB 11845986 IC50 = 21 nM T38763 C3X4VE 11845987 IC50 = 22 nM T38763 C3DUF6 11846504 IC50 = 200 nM T38763 C7QY0H 11847468 IC50 = 58 nM T38763 C7AUF4 11847469 IC50 = 69 nM T38763 CL0VW2 11847470 IC50 = 55 nM T38763 CHGF87 11847471 IC50 = 50 nM T38763 C28ZMC 11847472 IC50 = 16 nM T38763 C3P5TD 11987832 IC50 = 46 nM T38763 CZ6YJ7 11994755 IC50 = 26 nM T38763 C9LBU1 11994756 IC50 = 140 nM T38763 CQG3N9 11994883 IC50 = 140 nM T38763 C9GVA0 11994885 IC50 = 38 nM T38763 CKJZ05 11994886 IC50 = 19 nM T38763 CRJT15 11994887 IC50 = 26 nM T38763 CD0MO5 11994888 IC50 = 18 nM T38763 CAE62V 11994889 IC50 = 9 nM T38763 C1V7EH 11995124 IC50 = 21 nM T38763 C9I0UE 11995125 IC50 = 36 nM T38763 CBI7L8 11995126 IC50 = 41 nM T38763 COD10A 11995224 IC50 = 24 nM T38763 C6BAJ2 12292038 IC50 > 33000 nM T38763 CV2WN5 15877787 IC50 = 50000 nM T38763 CUB20Q 15949381 EC50 = 1100 nM T38763 C2GNV6 15954934 IC50 > 20000 nM T38763 CA7Q5R 15954935 IC50 > 20000 nM T38763 CA36YX 15954936 IC50 = 16300 nM T38763 CQZ3M8 15954937 IC50 = 1490 nM T38763 CVOT75 15954938 IC50 = 4460 nM T38763 CB0EK4 15955341 IC50 = 700 nM T38763 CNW94R 15955342 IC50 = 900 nM T38763 CN5X0T 15955343 IC50 = 900 nM T38763 CJDC52 15955344 IC50 = 1700 nM T38763 CIQ73O 15955345 IC50 = 1000 nM T38763 C70CTM 15955346 IC50 = 1200 nM T38763 CXLR02 15955347 IC50 = 2800 nM T38763 C21PMD 15955350 IC50 = 700 nM T38763 CRE1I4 15955351 IC50 = 3800 nM T38763 CIX7A6 15955352 IC50 = 4900 nM T38763 CF18ST 15955353 IC50 = 2000 nM T38763 CC45SR 15955354 IC50 = 500 nM T38763 C3L1EN 15955355 IC50 = 200 nM T38763 C8YQ1E 15955356 IC50 = 90 nM T38763 C4B6NE 15955357 IC50 = 500 nM T38763 CH9VU6 15955358 IC50 = 50 nM T38763 C3IT1J 15955359 IC50 = 150 nM T38763 C2XPA1 15955360 IC50 = 400 nM T38763 CV60HD 15955373 IC50 = 40 nM T38763 C4KVC6 15956742 IC50 = 1800 nM T38763 CT7R1G 15956743 IC50 = 4200 nM T38763 C6VF4E 15956782 IC50 = 390 nM T38763 CEL84W 15956783 EC50 = 1900 nM T38763 COP0D7 15956784 IC50 = 640 nM T38763 C51OVS 15956785 IC50 = 2200 nM T38763 C6FA5C 16072887 IC50 = 11200 nM T38763 CED6C1 16072888 IC50 = 77300 nM T38763 CKF86W 16072889 IC50 > 50000 nM T38763 CE54GA 16072890 IC50 = 4800 nM T38763 CSYQ10 16072892 IC50 = 94 nM T38763 C3HQ8V 16072893 IC50 = 1900 nM T38763 CP7SQ0 16072894 IC50 = 150 nM T38763 C6SIR9 16072895 IC50 = 320 nM T38763 CA0DK9 16074324 IC50 = 380 nM T38763 CQ1PK0 16075068 IC50 = 7900 nM T38763 CMP98J 16075069 IC50 = 1400 nM T38763 CVTI95 16075070 IC50 = 560 nM T38763 C6G9LX 16075071 IC50 = 2000 nM T38763 CV1CU2 16075072 IC50 = 7100 nM T38763 CY8D7I 16075073 IC50 = 1700 nM T38763 C5P2RG 16075074 IC50 = 240 nM T38763 CG5BI0 16076098 IC50 > 100000 nM T38763 C07IBX 16076099 IC50 = 93000 nM T38763 C9V7BR 16076100 IC50 = 52000 nM T38763 CWT13J 16076101 IC50 = 48000 nM T38763 C12AUT 16076102 IC50 = 9700 nM T38763 C0G8EV 16076103 IC50 = 2900 nM T38763 C07ZMS 16076104 IC50 = 1700 nM T38763 CNL35E 16076105 IC50 = 4300 nM T38763 C61UMZ 16076106 IC50 = 23000 nM T38763 CL9T7B 16076107 IC50 = 5000 nM T38763 CST82P 16076108 IC50 = 3600 nM T38763 CP39YN 16076109 IC50 = 1000 nM T38763 C3UAQ9 16076110 IC50 = 790 nM T38763 CPK29T 16076111 IC50 = 530 nM T38763 CFO6X7 16076181 IC50 = 44 nM T38763 CT3K9R 16631909 IC50 = 4797.33 nM T38763 CZW75X 16631912 IC50 = 84.92 nM T38763 CR9H8N 16631913 IC50 = 139.96 nM T38763 CK9B4J 16631984 IC50 = 139.96 nM T38763 CL89IN 16631988 IC50 = 279.9 nM T38763 C3IU0V 16632101 IC50 = 449.78 nM T38763 CSG04Z 16632104 IC50 = 779.83 nM T38763 CR8G7P 16632106 IC50 = 369.83 nM T38763 C2CJ0Z 16632107 IC50 = 389.94 nM T38763 CAG72H 18808412 IC50 = 34.99 nM T38763 C15TKE 18808457 IC50 = 2990 nM T38763 CW0YK3 18808489 IC50 = 1199.5 nM T38763 C1RXB9 18942298 IC50 = 2100 nM T38763 C8FBS9 21874515 IC50 = 180 nM T38763 C07JFR 22148303 IC50 = 4800 nM T38763 C0L2TF 23725128 IC50 = 96 nM T38763 CZFX47 24885633 IC50 = 280 nM T38763 C7LVW8 25014510 IC50 < 10000 nM T38763 CK3AF8 25256829 IC50 = 17000 nM T38763 COW8B1 44384615 IC50 = 2200 nM T38763 C2OY8Q 44384668 IC50 = 2900 nM T38763 CKI9L8 44385215 IC50 = 160 nM T38763 C2PMS8 44385644 IC50 = 60 nM T38763 CLK62H 44386091 IC50 = 400 nM T38763 C4Z8BA 44386386 IC50 = 1900 nM T38763 C06TWA 44386464 IC50 > 30000 nM T38763 CC49WM 44386485 IC50 = 1500 nM T38763 CP63VU 44386513 IC50 > 30000 nM T38763 C0M1CO 44386539 IC50 = 7000 nM T38763 CKI04C 44386563 IC50 > 30000 nM T38763 C2MT7E 44386694 IC50 > 30000 nM T38763 CP4JI6 44386743 IC50 > 30000 nM T38763 CNA64T 44386811 IC50 > 30000 nM T38763 CI7H4J 44386901 IC50 > 30000 nM T38763 CK6QV7 44386959 IC50 > 30000 nM T38763 CVON47 44387082 IC50 > 30000 nM T38763 CT18HB 44387140 IC50 > 30000 nM T38763 C87AXO 44387233 IC50 = 50000 nM T38763 CC5GX1 44387236 IC50 > 30000 nM T38763 C60WKU 44387237 IC50 > 30000 nM T38763 C3A9NB 44389500 IC50 = 310 nM T38763 CPA69U 44389502 IC50 = 1400 nM T38763 CYO91Q 44389996 IC50 = 400 nM T38763 CKBC05 44390013 IC50 = 700 nM T38763 CGLT15 44390034 IC50 > 20000 nM T38763 CT98RJ 44390075 IC50 = 18000 nM T38763 CL0IJ1 44390102 IC50 = 7600 nM T38763 CL92UP 44390117 IC50 = 12000 nM T38763 CSUT37 44391322 IC50 = 51000 nM T38763 CN2P7J 44391727 IC50 = 1600 nM T38763 CIJ0C8 44391954 IC50 = 5500 nM T38763 CT7RH3 44393278 IC50 = 2100 nM T38763 CAD71S 44393284 IC50 = 1400 nM T38763 CJCR94 44393307 IC50 = 910 nM T38763 CU3R8M 44393312 IC50 = 120 nM T38763 CZ6J2V 44393331 IC50 = 1300 nM T38763 C3YRL0 44393332 IC50 = 490 nM T38763 CVWT79 44393357 IC50 = 1200 nM T38763 CJ35RF 44393360 IC50 = 590 nM T38763 CH9P6F 44393384 IC50 > 10000 nM T38763 CCPU65 44398680 IC50 = 244 nM T38763 C2MSO0 44398715 IC50 = 13 nM T38763 CXMT85 44398743 IC50 = 78 nM T38763 C4FR5W 44398769 IC50 = 71 nM T38763 CON0W4 44399646 IC50 = 50 nM T38763 CZ8B7L 44400297 IC50 = 200 nM T38763 CYL8B5 44400509 IC50 = 2800 nM T38763 CL96RK 44400619 IC50 = 830 nM T38763 CV5YX2 44400808 IC50 = 13000 nM T38763 C7FWV8 44400819 IC50 = 790 nM T38763 C2D1EY 44400822 IC50 = 850 nM T38763 CL57SO 44400877 IC50 = 3100 nM T38763 CD67OZ 44400893 IC50 = 2200 nM T38763 C7UOR9 44400901 IC50 = 2000 nM T38763 CYJ96K 44400912 IC50 = 100 nM T38763 CW32OP 44404026 IC50 = 29000 nM T38763 C38RKF 44404032 IC50 = 68000 nM T38763 CY8V9Q 44404058 IC50 = 19000 nM T38763 CO3C2W 44404063 IC50 = 28000 nM T38763 CYP8V1 44404067 IC50 = 44000 nM T38763 CIT6P9 44404078 IC50 = 4000 nM T38763 CEV4T0 44406092 IC50 = 400 nM T38763 CZ3R9I 44406093 IC50 = 50 nM T38763 CZJ62A 44406100 IC50 = 50 nM T38763 CK2VS0 44406103 IC50 = 200 nM T38763 C5W8UT 44406118 IC50 = 200 nM T38763 C3RI7G 44406121 IC50 = 80 nM T38763 C5FJ9I 44406126 IC50 = 300 nM T38763 COES87 44406127 IC50 = 200 nM T38763 CAJ70H 44406137 IC50 = 500 nM T38763 CRM01D 44406145 IC50 = 300 nM T38763 CL0Q5Y 44406148 IC50 = 200 nM T38763 C5D6QF 44406149 IC50 = 600 nM T38763 C2YH3A 44406968 IC50 = 600 nM T38763 C9RH5Z 44406974 IC50 = 800 nM T38763 CAH5P2 44406992 IC50 = 6000 nM T38763 C35BWQ 44406993 IC50 = 500 nM T38763 CV60MI 44407003 IC50 = 700 nM T38763 C6MEA8 44407006 IC50 = 200 nM T38763 CY8PX1 44410817 IC50 > 33000 nM T38763 CGBF10 44410824 IC50 > 33000 nM T38763 CU16FT 44410825 IC50 > 33000 nM T38763 CZO5Q7 44410900 IC50 > 33000 nM T38763 CO8IF5 44411694 IC50 > 20000 nM T38763 CSJ6L5 44414040 IC50 > 50000 nM T38763 CRE6N9 44416835 IC50 = 820 nM T38763 CA06MQ 44416852 IC50 > 50000 nM T38763 CAYE41 44416853 IC50 > 100000 nM T38763 CY2NS0 44416893 IC50 = 75 nM T38763 C6TC1Z 44416908 IC50 = 340 nM T38763 CYF8X2 44416909 IC50 = 290 nM T38763 C5N3UL 44416926 IC50 = 480 nM T38763 CN4X9M 44417020 IC50 = 2200 nM T38763 C76FNI 44417042 IC50 = 81 nM T38763 C8GM2L 44417065 IC50 > 100000 nM T38763 C48WIT 44417164 IC50 = 5300 nM T38763 C06NJK 44417672 IC50 = 47 nM T38763 CALX92 44586007 IC50 = 25 nM T38763 COUC21 46878214 IC50 = 7600 nM T38763 CTPR49 46878215 IC50 = 6000 nM T38763 CD1R8O 46878216 IC50 = 5500 nM T38763 CCL42W 46898993 IC50 = 51.7 nM T38763 C16ZEM 46898994 IC50 = 24.4 nM T38763 CV0WS7 46905538 Ki = 229000 nM T38763 C2DCE0 46905539 Ki = 201000 nM T38763 CW0V2K 46905540 Ki = 327000 nM T38763 CAM4L7 49897232 IC50 = 439.54 nM T38763 CC3XK0 53318955 IC50 = 140 nM T38763 C09MWT 53373232 EC50 = 5 nM T38763 CY32HG 54677477 IC50 > 10000 nM T38763 CQ60PN 54704161 IC50 = 1000 nM T38763 C9ZKE7 54707373 IC50 = 80 nM T38763 CS93RI 54713196 IC50 = 930 nM T38763 CG6Y1O 54713243 IC50 = 69300 nM T38763 CZ4OQ7 54717319 IC50 = 8700 nM T38763 CM2G7P 54717321 IC50 = 79300 nM T38763 CW01IZ 54727422 IC50 > 100000 nM T38763 CWIG28 54727423 IC50 = 36000 nM T38763 CGJ3R2 54727893 IC50 = 4700 nM T38763 C9KN6A 56675170 IC50 = 150 nM T38763 C7VJ0F 57330244 EC50 = 26 nM T38763 C8Y4CZ 57330245 EC50 = 16 nM T38763 CS30XA 57330246 EC50 = 78 nM T38763 CRNV03 57330296 EC50 = 46 nM T38763 CM47IV 57330298 EC50 = 26 nM T38763 CW6G1F 57330299 EC50 = 11 nM T38763 CJE2L8 57330361 EC50 = 14 nM T38763 CDJ18M 57330421 EC50 = 43 nM T38763 CY34BS 57330425 EC50 = 56 nM T38763 CQL8D1 57330479 EC50 = 73 nM T38763 CTIK81 57330482 EC50 = 14 nM T38763 C1OIJ6 57330658 EC50 = 3 nM T38763 CL3GF9 57330659 EC50 = 4 nM T38763 CCP3U7 57330660 EC50 = 7 nM T38763 C7JZ8R 57330706 EC50 = 3 nM T38763 CN0PG6 57330707 EC50 = 8 nM T38763 CIK1G5 57330708 EC50 = 5 nM T38763 C2CE7B 57330760 EC50 = 9 nM T38763 CSEZ38 57330809 EC50 = 7 nM T38763 CJF9Q0 57330810 EC50 = 6 nM T38763 CI2WO9 57330866 EC50 = 3 nM T38763 C9WK0C 57330927 EC50 = 8 nM T38763 C5J4YT 57330988 EC50 = 7 nM T38763 CK24EM 57330990 EC50 = 74 nM T38763 C5CEZ0 57330992 EC50 = 5 nM T38763 CNZ10M 57331053 EC50 = 3 nM T38763 C5XHS4 57331054 EC50 = 3 nM T38763 CI5J7E 59233666 IC50 = 447 nM T38763 CQ0V8X 59275182 EC50 = 5.7 nM T38763 CEI1N4 59275359 EC50 = 3.8 nM T38763 C7GB2Q 59275584 EC50 = 22 nM T38763 CD6O7B 67719196 EC50 = 25 nM T38763 CCOG96 68063058 EC50 = 109 nM T38763 C1DLP0 68063060 EC50 = 182 nM T38763 CRH94E 68063519 EC50 = 24 nM T38763 CWAJ16 68063521 EC50 = 1208 nM T38763 CYNF16 69191005 EC50 = 59 nM T38763 C9H1YR 69191011 EC50 = 13 nM T38763 CD68XU 69191034 EC50 = 13 nM T38763 CX96IE 69191037 EC50 = 666 nM T38763 CP1AY0 69191041 EC50 = 19 nM T38763 C64DVR 69191527 EC50 = 164 nM T38763 CHI9D6 69191553 EC50 = 451 nM T38763 CMH5R7 69192002 EC50 = 5 nM T38763 C7PHI2 69192762 EC50 = 38 nM T38763 C2IO5E 70800540 EC50 = 20 nM T38763 C2CT0V 70800543 EC50 = 17 nM T38763 CSY2I5 70800548 EC50 = 107 nM T38763 CBC72P 70800558 EC50 = 304 nM T38763 CP1Z2A 70800628 EC50 = 11 nM T38763 CX28FO 70800716 EC50 = 686 nM T38763 C37WZV 70800722 EC50 = 850 nM T38763 CLBT35 70800757 EC50 > 2000 nM T38763 C3QZ7G 70800831 EC50 = 17 nM T38763 CL58OW 70800833 EC50 = 15 nM T38763 CAL0W4 70800848 EC50 = 12 nM T38763 C2E4AM 70800857 EC50 = 586 nM T38763 C1PZ3V 70800859 EC50 = 1473 nM T38763 CFYI23 70800865 EC50 = 69 nM T38763 CVZJ57 70800869 EC50 = 33 nM T38763 C34JPC 70800874 EC50 = 19 nM T38763 CISF49 70800914 EC50 = 13 nM T38763 CG34FW 70800921 EC50 = 13 nM T38763 C9A0NX 71263595 EC50 = 2.2 nM T38763 CWS95U 71263604 EC50 = 0.9 nM T38763 CQSU48 71263605 EC50 = 1.1 nM T38763 C9AT8D 71263621 EC50 = 1.2 nM T38763 CT9QU8 71263635 EC50 = 1 nM T38763 CFA9V1 71494937 EC50 = 1.3 nM T38763 C1DF4I 71509114 EC50 = 1.1 nM T38763 CC1XQ3 73345768 IC50 = 310 nM T38763 CWM9P6 73345770 IC50 = 3200 nM T38763 C6FQ0B 73347254 IC50 = 2000 nM T38763 COUR90 73351864 IC50 > 10000 nM T38763 C0UX3I 73891124 IC50 = 90 nM T38763 C40FLD 73891125 IC50 = 27 nM T38763 CEJ43L 75250792 IC50 = 0.001 nM T38763 CTOE72 76283266 IC50 = 54000 nM T38763 CI20UY 76286118 IC50 = 140 nM T38763 CVGU57 76286400 IC50 = 39 nM T38763 CS2M5X 76286401 IC50 = 860 nM T38763 CU0F1P 76286540 IC50 = 110 nM T38763 C83NXO 76286544 IC50 = 340 nM T38763 CCI51H 76286694 IC50 = 6400 nM T38763 CHL7Z6 76286696 IC50 = 84000 nM T38763 CI0Q4F 76287000 IC50 = 150 nM T38763 CH8C0I 76310816 Ki = 130 nM T38763 C34TAM 77845572 EC50 = 0.86 nM T38763 C2NCH9 78318214 EC50 = 0.63 nM T38763 C2GET7 78318815 EC50 = 0.9 nM T38763 C16KHY 85470079 IC50 = 9.6 nM T38763 C7WS8R 85470298 IC50 = 15 nM T38763 C23HQZ 85471415 IC50 = 9 nM T38763 CV6NO1 85472072 IC50 = 6 nM T38763 CGCB62 85473348 IC50 = 15 nM T38763 C3MXE8 85473349 IC50 = 32 nM T38763 CE50VY 85473351 IC50 = 17 nM T38763 CQ9P5W 88576864 EC50 = 298 nM T38763 C15ZLQ 88981488 EC50 = 31 nM T38763 CK8Y7B 90332545 EC50 = 2.2 nM T38763 C9IA2N 90333582 EC50 = 1.9 nM T38763 CCKA85 90333844 EC50 = 1.1 nM T38763 C26LKW 90341025 EC50 = 0.95 nM T38763 CCV92Z 98207021 IC50 = 3531.83 nM T38763 C3RCP8 117775248 EC50 = 0.61 nM T38763 CU4G2C 117940941 IC50 = 300 nM T38763 CAE1S4 118468989 EC50 = 4000 nM T38763 C65XGZ 118524955 IC50 = 10 nM T38763 CE83WQ 124220774 IC50 = 16 nM T38763 CJY2C8 127041823 EC50 > 50000 nM T38763 C3TC9O 134828054 EC50 = 5.4 nM T38763 CSYU89 135399778 IC50 > 10000 nM T38763 CW2YT7 135399779 IC50 = 81 nM T38763 CLRG32 135403095 IC50 > 10000 nM T38763 C6N3RO 135403096 IC50 > 10000 nM T38763 C29BMF 135403097 IC50 = 108 nM T38763 CP5G7U 135406878 IC50 = 2300 nM T38763 C8O1QZ 135406950 IC50 = 1600 nM T38763 C80KUQ 135409287 IC50 = 4000 nM T38763 CZ9IP2 135410230 IC50 = 600 nM T38763 CCN19W 135410964 IC50 = 63 nM T38763 C7L8TH 135410965 IC50 = 189 nM T38763 C4B7UJ 135410966 IC50 = 88 nM T38763 CYDF29 135410967 IC50 = 72 nM T38763 CT40BH 135410968 IC50 = 6.7 nM T38763 CWI4E7 135410969 IC50 = 58 nM T38763 CZM4K9 135410970 IC50 = 21 nM T38763 CN80KH 135410971 IC50 = 61 nM T38763 CGB35E 135410972 IC50 = 87 nM T38763 C70LIM 135410973 IC50 = 96 nM T38763 C5IL8G 135410974 IC50 = 50 nM T38763 CW7XR2 135410975 IC50 = 48 nM T38763 C54ZYL 135410976 IC50 = 20 nM T38763 C06BQT 135410977 IC50 = 43 nM T38763 C61WDB 135410978 IC50 = 18 nM T38763 C2XT8I 135410979 IC50 = 132 nM T38763 CB89IW 135410980 IC50 = 115 nM T38763 C28BHN 135410981 IC50 = 43 nM T38763 C4U8LE 135410982 IC50 = 43 nM T38763 CPRM96 135410983 IC50 = 129 nM T38763 C1QZE4 135410984 IC50 = 18 nM T38763 C4WYA9 135410985 IC50 = 5.5 nM T38763 CZ7CK4 135410986 IC50 = 41 nM T38763 CFJP26 135410987 IC50 = 107 nM T38763 C2D1HF 135410988 IC50 = 67 nM T38763 COH3X5 135410989 IC50 = 39 nM T38763 CNER49 135410990 IC50 = 10 nM T38763 C2MEH6 135410992 IC50 = 20 nM T38763 CFZ6K9 135410993 IC50 = 10 nM T38763 CR9Z4J 135410994 IC50 = 15 nM T38763 CA1IN5 135410995 IC50 = 57 nM T38763 C71TBG 135410996 IC50 = 13 nM T38763 C9Q5IG 135411000 IC50 = 121 nM T38763 CWB0N1 135411001 IC50 = 2.8 nM T38763 CC8S1R 135411002 IC50 = 14 nM T38763 C6TNQ8 135412361 EC50 = 417 nM T38763 CKD6C1 135414267 IC50 = 24 nM T38763 CX9FQ3 135414349 IC50 > 50000 nM T38763 CTU68D 135414351 IC50 = 240 nM T38763 C9BES8 135414358 IC50 = 2400 nM T38763 CJU4E1 135414492 IC50 = 280 nM T38763 C5HV2A 135415565 EC50 > 50000 nM T38763 C1HLR6 135421250 IC50 = 500 nM T38763 C36AWG 135421265 IC50 = 1.4 nM T38763 CJB59I 135421310 EC50 = 152 nM T38763 CAG9V5 135421576 IC50 = 5592 nM T38763 C1E2BF 135424684 IC50 > 10000 nM T38763 CB2W3T 135424698 IC50 > 10000 nM T38763 CDVX06 135424720 IC50 > 10000 nM T38763 CG3OX6 135425215 IC50 = 290 nM T38763 CVA01C 135425222 IC50 = 620 nM T38763 CNAB36 135425226 IC50 = 41 nM T38763 CC9Q7J 135425229 IC50 = 528 nM T38763 C8SUN6 135425247 IC50 = 316 nM T38763 C2SMJ4 135427888 IC50 = 5300 nM T38763 CP87WO 135427952 IC50 = 800 nM T38763 C7THV3 135428011 IC50 > 10000 nM T38763 CB5XE1 135430344 IC50 = 1490 nM T38763 C3YX5Z 135430587 IC50 = 6200 nM T38763 C8DW6P 135430590 IC50 = 2220 nM T38763 C4PD7N 135430710 IC50 = 23 nM T38763 CNP81S 135433053 IC50 = 1550 nM T38763 CLB7J2 135433098 IC50 = 179 nM T38763 CSA8P6 135433129 IC50 = 65 nM T38763 CE9X0V 135433415 IC50 = 240 nM T38763 C2GOX3 135433495 IC50 = 130 nM T38763 CV8LP6 135434352 IC50 = 15000 nM T38763 C4QHN2 135434387 IC50 = 1400 nM T38763 C53AWL 135434400 IC50 = 44 nM T38763 C7IH2F 135434403 IC50 = 90 nM T38763 CY9E0C 135434404 IC50 = 200 nM T38763 C83VZI 135434405 IC50 = 230 nM T38763 CF5S2L 135434406 EC50 = 31500 nM T38763 C5T0CY 135434413 EC50 = 18600 nM T38763 C0QB8N 135434414 EC50 = 13600 nM T38763 CO42SE 135434417 IC50 = 380 nM T38763 CANC32 135434418 IC50 = 220 nM T38763 C67YHU 135434420 IC50 = 460 nM T38763 C9L3KG 135434428 IC50 = 230 nM T38763 C0PV2O 135434430 IC50 = 210 nM T38763 C3Y4BS 135434464 IC50 = 580 nM T38763 CVY7C1 135434466 IC50 = 580 nM T38763 C3FL8E 135434518 IC50 = 1420 nM T38763 C0ER9H 135434542 IC50 = 1900 nM T38763 C5EKV3 135434570 IC50 = 5600 nM T38763 C08FMK 135434616 IC50 = 9400 nM T38763 CZ72WN 135434617 IC50 = 13800 nM T38763 CYC68B 135434620 IC50 = 16000 nM T38763 COQ8T1 135434622 IC50 = 48600 nM T38763 CH9EM8 135434623 IC50 = 11600 nM T38763 C8G3PC 135434747 IC50 = 2770 nM T38763 CS9U6W 135435179 IC50 = 30000 nM T38763 CG6O1A 135435180 IC50 > 50000 nM T38763 C63ONQ 135435181 IC50 = 13 nM T38763 CO9ET5 135435182 IC50 = 15000 nM T38763 CV65JE 135435183 IC50 > 100000 nM T38763 CVN2O6 135435184 IC50 > 100000 nM T38763 CKSD39 135435185 IC50 = 3000 nM T38763 CQA85B 135435186 IC50 > 100000 nM T38763 C56ELQ 135435187 IC50 = 23000 nM T38763 CFB25U 135435188 IC50 = 30000 nM T38763 C5Z4CL 135435189 IC50 > 100000 nM T38763 CML2T3 135435190 IC50 > 100000 nM T38763 C8JC6V 135438359 EC50 = 298 nM T38763 CW7KD5 135438546 IC50 > 10000 nM T38763 C0FXB6 135438563 IC50 = 4328 nM T38763 C0IAM8 135441196 IC50 = 2 nM T38763 C5ZD7G 135444726 IC50 = 42 nM T38763 CZ4GP6 135446244 IC50 > 10000 nM T38763 CFE08I 135446989 IC50 > 10000 nM T38763 CZO16E 135446990 IC50 = 696 nM T38763 CA7T8B 135449954 IC50 = 289 nM T38763 C9W6DI 135449992 EC50 = 274 nM T38763 CQ9YR3 135449994 IC50 = 82 nM T38763 C0QRI4 135449998 IC50 = 340 nM T38763 CS9JC7 135450035 IC50 > 10000 nM T38763 CUO9W5 135450089 EC50 = 370 nM T38763 C7FA0I 135450101 IC50 = 144 nM T38763 CADN68 135450136 IC50 = 3950 nM T38763 C5GY7R 135452833 IC50 = 455 nM T38763 CSG69E 135453121 IC50 = 338 nM T38763 CG51RY 135453371 IC50 = 118 nM T38763 CL7W1M 135453408 IC50 = 80 nM T38763 C4HCU6 135453429 IC50 = 484 nM T38763 CJ0QV4 135453432 IC50 = 21 nM T38763 CFAS97 135453441 IC50 = 554 nM T38763 CH3O0K 135453452 IC50 = 367 nM T38763 CED23H 135453464 EC50 = 1204 nM T38763 CGCM84 135457065 IC50 > 10000 nM T38763 C90UXV 135458461 IC50 = 5.2 nM T38763 CX1UJ8 135461093 IC50 > 10000 nM T38763 C05IWT 135464356 IC50 = 93 nM T38763 C04DHY 135465480 IC50 > 25000 nM T38763 C3S6XO 135465481 IC50 > 50000 nM T38763 CL3T1U 135465482 IC50 = 680 nM T38763 C5K1ZV 135466575 IC50 > 10000 nM T38763 C2P7BL 135467940 IC50 = 6503 nM T38763 CUW92K 135469509 IC50 = 2036 nM T38763 CRXT07 135469523 IC50 = 132 nM T38763 C1QVX0 135469533 IC50 = 2537 nM T38763 CW9S6H 135469558 IC50 = 33 nM T38763 C8NHV5 135469562 IC50 = 2322 nM T38763 CIW3N1 135469610 IC50 = 290 nM T38763 CIBZ50 135473606 IC50 > 100000 nM T38763 C8H3WJ 135474724 IC50 = 3900 nM T38763 C5GNH4 135474766 IC50 = 1170 nM T38763 CY3K9S 135477944 IC50 = 3 nM T38763 CDSY07 135485553 IC50 = 20500 nM T38763 CHVM59 135485658 IC50 = 70 nM T38763 CDR1S6 135487401 IC50 = 95 nM T38763 CQ63UC 135489353 IC50 > 2429 nM T38763 CEXM45 135489371 IC50 > 10000 nM T38763 CS8DC6 135489390 IC50 = 2442 nM T38763 CQPB87 135489397 IC50 > 10000 nM T38763 C1HWP4 135489541 IC50 > 10000 nM T38763 C0RPE8 135491787 IC50 > 10000 nM T38763 CHD5C4 135491920 IC50 > 10000 nM T38763 CTQD64 135494585 IC50 = 810 nM T38763 C5ROC8 135500123 IC50 = 58 nM T38763 CLPO83 135502999 IC50 = 819 nM T38763 C7KF4D 135503019 IC50 > 10000 nM T38763 CS0U5I 135503040 IC50 = 1741 nM T38763 C9K2JL 135503052 IC50 = 36 nM T38763 C23TUF 135505666 IC50 > 10000 nM T38763 CI69VO 135505680 IC50 > 10000 nM T38763 CX7UN9 135505824 IC50 = 1035 nM T38763 CGPH04 135507319 IC50 = 16750 nM T38763 CLA5M9 135510005 IC50 = 47 nM T38763 CHA21P 135510013 IC50 = 780 nM T38763 C07ZXH 135510016 IC50 > 10000 nM T38763 CL4A2J 135513149 IC50 > 10000 nM T38763 CAY16J 135513163 IC50 = 90 nM T38763 C3IOW6 135517454 IC50 = 83 nM T38763 C7GKJ0 135519524 EC50 = 444 nM T38763 CHSG18 135520480 IC50 = 2815 nM T38763 CRGB28 135520489 IC50 > 10000 nM T38763 CZ1V6S 135524693 IC50 = 13200 nM T38763 C3XUY1 135524694 IC50 = 50000 nM T38763 C8SF3M 135524695 IC50 = 58000 nM T38763 C49SWT 135525394 IC50 = 230 nM T38763 CP63YL 135525568 IC50 > 10000 nM T38763 C9FOJ6 135525573 IC50 > 10000 nM T38763 C4TAD3 135525592 IC50 = 61 nM T38763 CP14ZI 135527125 IC50 = 150 nM T38763 C4C5LY 135529534 EC50 = 241 nM T38763 CG4BQ5 135530111 EC50 = 774 nM T38763 CDRZ58 135530124 IC50 = 304 nM T38763 CYU2H5 135530132 IC50 = 21 nM T38763 CK1PQ7 135530445 EC50 = 389 nM T38763 C8G7ZA 135530447 IC50 = 750 nM T38763 C1RD0A 135530454 EC50 = 157 nM T38763 CN9Q7C 135530457 IC50 = 206 nM T38763 CS6A0Y 135530458 IC50 = 47 nM T38763 CM37PF 135530473 IC50 = 20 nM T38763 CDL6O3 135530514 IC50 = 106 nM T38763 CKOJ95 135530515 IC50 > 10000 nM T38763 CDJ2Y8 135530577 IC50 = 105 nM T38763 CAO52J 135530699 IC50 = 5805 nM T38763 CG1AO2 135530708 IC50 = 973 nM T38763 C5FB9T 135530714 IC50 = 4235 nM T38763 C13HMB 135532469 IC50 = 78 nM T38763 CRYV96 135532470 IC50 = 90 nM T38763 CI8U1S 135532507 IC50 = 1301 nM T38763 C6CRK9 135532542 IC50 = 198 nM T38763 C0VY3Q 135532713 IC50 = 1800 nM T38763 CA7DL8 135532809 IC50 = 82 nM T38763 CI3V7M 135532828 IC50 = 23 nM T38763 C5SMA1 135532856 IC50 = 44 nM T38763 CR9PN0 135537607 IC50 = 96 nM T38763 C8C4VX 135541370 IC50 = 2120 nM T38763 CUP59V 135541371 IC50 = 8310 nM T38763 CB9P5L 135541372 IC50 = 54 nM T38763 CNU4B8 135541373 IC50 = 2510 nM T38763 CG6X1J 135541374 IC50 = 1170 nM T38763 C4CXG6 135541375 IC50 = 65 nM T38763 CXSN12 135541376 IC50 = 930 nM T38763 C6ZIN0 135541377 IC50 = 1490 nM T38763 C4GAX8 135541378 IC50 = 850 nM T38763 C1FUY5 135541379 IC50 = 367 nM T38763 C5KTH2 135541380 IC50 = 80 nM T38763 CUIJ64 135541381 IC50 = 46 nM T38763 C2XVZ0 135541382 IC50 = 51 nM T38763 C1JL6K 135541383 IC50 = 25 nM T38763 C4BXK7 135541384 IC50 = 24 nM T38763 CO17TZ 135541385 IC50 = 34 nM T38763 C7B2KF 135541386 IC50 = 906 nM T38763 C3AP2N 135541387 IC50 = 41 nM T38763 C4M0DW 135541388 IC50 = 3 nM T38763 CCS0E1 135541389 IC50 = 5 nM T38763 C96HKU 135542915 IC50 = 172 nM T38763 C04YKD 135542929 IC50 = 53 nM T38763 C3XJE4 135542946 IC50 = 2694 nM T38763 C7Q5SL 135543039 IC50 = 205 nM T38763 COJ26C 135545831 IC50 > 10000 nM T38763 C4S6IF 135546397 IC50 = 20000 nM T38763 C1YM4E 135547941 EC50 = 265 nM T38763 C7NHZ3 135905448 IC50 = 253.8 nM T38763 CD91OI 136029175 IC50 > 30000 nM T38763 CUX2B1 136043747 IC50 = 24 nM T38763 C8SZX6 136043752 IC50 = 32 nM T38763 C57QLR 136043760 IC50 = 8.7 nM T38763 CI8Y1F 136043763 IC50 = 51 nM T38763 CX7O3N 136043775 IC50 = 27 nM T38763 CCDA54 136048750 IC50 > 100000 nM T38763 CX9VH3 136048751 IC50 = 58000 nM T38763 CJU90V 136048767 IC50 = 135 nM T38763 CR31XE 136048768 IC50 = 108 nM T38763 CH27SJ 136048769 IC50 = 129 nM T38763 CBN5Q2 136048770 IC50 = 6720 nM T38763 CSWM10 136048771 IC50 = 951 nM T38763 C7GB4U 136048772 IC50 = 1490 nM T38763 C6LO4X 136048773 IC50 > 5000 nM T38763 CUW07Y 136048774 IC50 = 134 nM T38763 C6PHE0 136048775 EC50 = 1350 nM T38763 CNH10V 136048776 IC50 = 75 nM T38763 C7CU5A 136048777 IC50 = 4690 nM T38763 C0VK8B 136048778 IC50 = 439 nM T38763 C4N9VK 136048779 IC50 = 481 nM T38763 C97ZOY 136048780 EC50 = 1050 nM T38763 C1TG7Y 136048781 IC50 = 150 nM T38763 C50UYZ 136048782 IC50 = 928 nM T38763 C0G2EB 136048783 IC50 = 212 nM T38763 CUP8F3 136048784 IC50 = 125 nM T38763 CPM81H 136048785 IC50 = 1450 nM T38763 C9FLK8 136048786 IC50 = 674 nM T38763 C3DH4O 136048787 IC50 = 217 nM T38763 CDF9V0 136048788 IC50 = 1130 nM T38763 CA1JS8 136048789 IC50 = 1800 nM T38763 CB81YW 136048790 IC50 = 386 nM T38763 C5Y0FT 136048791 IC50 = 1190 nM T38763 C6O2ES 136048792 IC50 = 221 nM T38763 C8BKU0 136048793 IC50 = 305 nM T38763 C4G1YH 136048794 IC50 = 4630 nM T38763 CK3UO6 136048795 IC50 = 133 nM T38763 C15YDK 136048796 IC50 = 150 nM T38763 C4YNM5 136048797 IC50 = 120 nM T38763 C85LOE 136048798 IC50 = 6350 nM T38763 CUWP73 136196524 IC50 = 60 nM T38763 CUVF07 136224043 IC50 = 21000 nM T38763 CP0J3S 136224044 IC50 = 57000 nM T38763 CVM8U1 136224045 IC50 = 13000 nM T38763 CN84SV 136224046 IC50 = 22000 nM T38763 CG8NO0 136224047 IC50 = 20000 nM T38763 C43OTF 136224048 IC50 = 8600 nM T38763 C52EXZ 136224049 IC50 = 9200 nM T38763 C4PV3D 136224050 IC50 = 3800 nM T38763 C6SQ4R 136224274 IC50 = 30000 nM T38763 C5IY9Q 136224275 IC50 = 7100 nM T38763 C14ONV 136224276 IC50 = 13000 nM T38763 CRFG35 136224277 IC50 = 37153.52 nM T38763 C20SBI 136224278 IC50 = 15000 nM T38763 C1FD8L 136224279 IC50 = 27000 nM T38763 CX83VJ 136224280 IC50 = 25118.86 nM T38763 C96OYA 136224281 IC50 = 50000 nM T38763 CYAJ67 136224282 IC50 = 12882.5 nM T38763 C7IPY9 136240154 IC50 = 12022.64 nM T38763 C8BTY2 136240155 IC50 = 10000 nM T38763 C2AP5U 136240156 IC50 = 13000 nM T38763 CUT67N 136240157 IC50 = 30000 nM T38763 C0CB8K 136240158 IC50 = 18197.01 nM T38763 CZ5W8L 136240166 IC50 = 33113.11 nM T38763 CEY3H7 136241493 IC50 = 32000 nM T38763 C0BZ3C 136241494 IC50 = 11000 nM T38763 C1FAB0 136241495 IC50 = 12000 nM T38763 C7XWF2 136241496 IC50 = 29000 nM T38763 CR6I9J 136241497 IC50 = 12000 nM T38763 CH8R3E 136245148 IC50 = 11000 nM T38763 CT79WY 136245149 IC50 = 14000 nM T38763 CR1Y7I 136245150 IC50 = 12022.64 nM T38763 CF81GW 136245151 IC50 = 18000 nM T38763 C5E2JM 136245152 IC50 = 19952.62 nM T38763 CC54BK 136245157 IC50 = 11000 nM T38763 C46IUL 136249249 IC50 = 25000 nM T38763 CWK6E5 136249250 IC50 = 12000 nM T38763 CPI8W1 136249251 IC50 = 19000 nM T38763 CXQV80 136249252 IC50 = 14000 nM T38763 CUJ3B1 136249253 IC50 = 9900 nM T38763 CN1AL0 136249254 IC50 = 16982.44 nM T38763 CP7SZ0 136260029 IC50 = 16982.44 nM T38763 C3C9XE 136260032 IC50 = 10000 nM T38763 C94VKX 136260042 IC50 = 14000 nM T38763 CG8D7A 136260043 IC50 = 34000 nM T38763 C2F1GO 136260046 IC50 = 12022.64 nM T38763 C1SEH4 136260047 IC50 = 10964.78 nM T38763 CA6N7O 136260050 IC50 = 34000 nM T38763 C3L7KP 136260051 IC50 = 8700 nM T38763 C7E2UJ 136260059 IC50 = 14000 nM T38763 CY74LK 136264332 IC50 = 32000 nM T38763 CDNV51 139030268 EC50 = 2 nM T38763 C1BOT2 139030270 EC50 = 1.1 nM T38763 C6NL8U 145961743 IC50 = 330 nM T38763 C7TUZ3 145964167 IC50 = 9900 nM T38763 CE25KX 145964855 IC50 = 1100 nM T38763 C89YWK 145967607 EC50 = 34.52 nM T38763 CYJ3I2 145967634 EC50 = 52.34 nM T38763 CMF61R 145968299 EC50 = 93.46 nM T38763 CKH2P0 145968901 EC50 = 83.75 nM T38763 CFG75P 145969527 EC50 = 96.35 nM T38763 C5BNT8 145970805 EC50 = 37.03 nM T38763 CFVW25 145970962 EC50 = 22.83 nM T38763 C8N1EK 145971048 EC50 = 12.64 nM T38763 CPT3Q4 145972846 IC50 = 3600 nM T38763 CF7GA4 145976581 IC50 = 430 nM T38763 C1INU3 145977099 IC50 = 160 nM T38763 CHO6Y4 145978981 IC50 = 11 nM T38763 CKX3M5 145979083 IC50 = 7943.28 nM T38763 CRM5H7 145979956 IC50 = 61 nM T38763 C4KXC8 145980451 IC50 = 50 nM T38763 CH4F0U 145980805 IC50 = 35 nM T38763 CP29DO 145982313 IC50 = 362 nM T38763 CW4AT8 145982334 IC50 = 64 nM T38763 C38RHZ 145984139 IC50 = 96 nM T38763 CH4XF2 145986389 IC50 = 99 nM T38763 CX43CP 145986494 IC50 = 5 nM T38763 C7YLS1 145986525 IC50 = 43 nM T38763 CG1PV7 145987277 EC50 = 1.163 nM T38763 CJ3UP2 145987631 IC50 = 6309.57 nM T38763 CLE4I6 145987724 EC50 = 21.36 nM T38763 CX8B0D 145987946 EC50 = 18.32 nM T38763 CX0G7R 145988767 IC50 = 630.96 nM T38763 CBC7K2 145989542 IC50 = 2511.89 nM T38763 C98UQL 145989571 IC50 = 5 nM T38763 C2JUQ6 145989797 IC50 = 305 nM T38763 C5AB9N 145990068 IC50 = 66 nM T38763 CTGS04 145990397 IC50 = 20 nM T38763 CT0GQ2 145990654 IC50 = 27 nM T38763 CD54GH 145991001 IC50 = 18 nM T38763 CY4DZ5 145991112 IC50 = 18 nM T38763 C4YAL3 145991203 IC50 = 501.19 nM T38763 C4QAI9 145991419 IC50 = 10 nM T38763 CTW8R1 145992676 IC50 = 31 nM T38763 COT6K2 145993037 IC50 = 3162.28 nM T38763 CL8ND6 145993567 IC50 = 187 nM T38763 CG50ZK 145993705 IC50 = 17 nM T38763 C6A3BJ 155510584 EC50 = 50 nM T38763 COL3R6 155511228 EC50 = 15000 nM T38763 C1Y3GO 155512686 IC50 = 1370 nM T38763 CT74QE 155513632 EC50 = 2.3 nM T38763 CJ8BT7 155514121 IC50 = 220 nM T38763 CMZE38 155514266 EC50 = 15 nM T38763 CD3BW6 155516165 IC50 = 1260 nM T38763 CT5SA0 155516365 EC50 = 600 nM T38763 C16EHK 155516673 EC50 = 250 nM T38763 C03YKV 155518249 EC50 = 13 nM T38763 C4RD5M 155518440 IC50 = 5116.82 nM T38763 CC83NX 155519484 IC50 = 90 nM T38763 CW46LE 155520559 EC50 = 1.2 nM T38763 CI8P7T 155521578 EC50 = 28 nM T38763 CLA97W 155522113 IC50 = 69.98 nM T38763 C4NS1O 155522949 EC50 = 60000 nM T38763 C7A1IX 155523552 EC50 > 10000 nM T38763 CVA8H7 155524476 EC50 = 21 nM T38763 C4HEK5 155527957 EC50 = 9.2 nM T38763 C37GZH 155528032 EC50 = 3.8 nM T38763 CF0O1G 155529099 EC50 = 500 nM T38763 C6EV2O 155529280 IC50 = 319.89 nM T38763 CAL84B 155530316 IC50 = 760 nM T38763 CH0F2W 155532431 EC50 = 290 nM T38763 CWO5N3 155532638 EC50 = 45000 nM T38763 CP8BE2 155533543 EC50 = 3.4 nM T38763 CWX93D 155533768 EC50 = 16 nM T38763 CZ3DW6 155533821 EC50 = 120 nM T38763 CC9ND2 155534918 EC50 = 140 nM T38763 CZA90U 155535017 EC50 = 7500 nM T38763 CAW0G5 155535026 IC50 = 196.6 nM T38763 CN3P9H 155537022 EC50 = 8.3 nM T38763 CJ2Z7X 155537035 EC50 = 6 nM T38763 CCF12Y 155537239 EC50 = 9 nM T38763 C4QO5G 155538369 EC50 = 40000 nM T38763 CWAQ10 155539975 EC50 = 15000 nM T38763 CSV87B 155542372 IC50 = 199.99 nM T38763 CLC1V0 155542404 EC50 = 30000 nM T38763 CE18OX 155544504 EC50 = 7000 nM T38763 CQ4MD8 155545029 EC50 = 30000 nM T38763 C7UW8D 155545588 EC50 = 2000 nM T38763 CUN65L 155546880 EC50 = 1.2 nM T38763 CJNZ71 155547419 EC50 = 600 nM T38763 C7C0FQ 155550131 EC50 = 600 nM T38763 CM93UW 155550449 EC50 = 20 nM T38763 C9I8RV 155552218 EC50 = 35 nM T38763 CG1S0K 155552808 IC50 = 75.3 nM T38763 CWS7I2 155552926 EC50 = 11 nM T38763 CJ82IN 155553685 EC50 = 6.6 nM T38763 CVF8Q0 155553708 EC50 > 10000 nM T38763 CI90NU 155554296 IC50 = 430.8 nM T38763 C6NCH4 155554702 EC50 = 2000 nM T38763 CRC1S8 155554973 EC50 = 60000 nM T38763 CJQG41 155558439 IC50 = 2197.86 nM T38763 C5DNJ9 155561940 EC50 = 8.8 nM T38763 CTF43C 155562565 EC50 = 165 nM T38763 CHR09Q 155564800 EC50 = 7100 nM T38763 C6SY7F 155565358 IC50 = 539.51 nM T38763 CY6HV1 155565523 IC50 = 429.54 nM T38763 CA12YD 155567103 EC50 = 100000 nM T38763 C1T4JN 155567349 EC50 = 18 nM T38763 C1DHM3 155567354 EC50 = 63 nM T38763 COY5W6 155568636 EC50 = 100 nM T38763 C6W3NG 155569058 IC50 = 190 nM T38763 D0J0HK 135440068 IC50 = 600 nM T38763 D0Q9MA 6303 IC50 = 22000 nM T80423 D0Q2SE 56684144 IC50 = 4100 nM T80423 CI70QW 66545747 IC50 = 900 nM T80423 C9H7GQ 91799297 IC50 = 656 nM T76914 D09GOS 2812 IC50 = 6000 nM T76914 D0J2TN 13505 IC50 = 5000 nM T76914 D0R0FE 2520 IC50 = 8000 nM T76914 D0QR5G 2355 IC50 = 101000 nM T76914 D0G1VS 656768 IC50 = 200 nM T76914 CI14YT 137944 IC50 = 20000 nM T76914 C8XDI4 224577 IC50 = 20500 nM T76914 CO8JK1 605100 IC50 = 1860 nM T76914 CYO4C2 641785 IC50 = 2 nM T76914 CPDZ17 3718350 IC50 = 1030 nM T76914 CP4ZT3 3941392 IC50 = 5010 nM T76914 CSPK30 5348558 EC50 = 400 nM T76914 C6HA8E 5388709 IC50 > 30000 nM T76914 C8W2QA 6439099 IC50 = 2500 nM T76914 CEY50T 6918568 IC50 = 3900 nM T76914 COKI25 9796735 IC50 = 544 nM T76914 COT0M7 9804657 IC50 = 1270 nM T76914 CG1DH8 9847973 IC50 = 500 nM T76914 CKXO76 9884639 EC50 = 1000 nM T76914 CMNO90 9974422 IC50 = 65 nM T76914 C2U9SP 9977230 IC50 = 88 nM T76914 CGC07F 10030698 IC50 = 2900 nM T76914 CSI6R8 10089473 EC50 = 800 nM T76914 C5IC3J 10113124 IC50 = 5 nM T76914 C7GMX4 10137057 IC50 = 18 nM T76914 C48ILP 10137280 IC50 = 140 nM T76914 CYUK76 10178880 IC50 = 5 nM T76914 C2CQF5 10245349 IC50 > 5000 nM T76914 CT9Y6V 10247467 IC50 = 471 nM T76914 CR2ZB1 10248488 IC50 = 275 nM T76914 CJ95LE 10250802 IC50 = 213 nM T76914 C0SA1P 10252803 IC50 = 75 nM T76914 CSHY35 10268705 IC50 = 200 nM T76914 CQF1C8 10315748 IC50 = 47 nM T76914 CVM3P6 10338126 IC50 = 32 nM T76914 C2KIL3 10387528 IC50 = 72 nM T76914 CX42UJ 10405481 IC50 = 475 nM T76914 CZ1D4R 10428385 IC50 = 227 nM T76914 CU4J8Y 10431492 IC50 = 239 nM T76914 C0JX1Y 10596590 IC50 > 30000 nM T76914 CZTW32 11403645 EC50 = 17000 nM T76914 C03PJA 11652981 IC50 = 5000 nM T76914 CLV7M9 11742533 IC50 = 240 nM T76914 CI6WQ5 12300622 IC50 = 1700 nM T76914 C8GCV7 16280560 IC50 > 30000 nM T76914 C53KWD 18009422 IC50 = 7200 nM T76914 CJR83C 18009423 IC50 = 29 nM T76914 CNI6B0 18009426 IC50 = 130 nM T76914 COX83C 18009437 IC50 = 140 nM T76914 CE27FW 18009438 IC50 = 3730 nM T76914 CZD8B4 18009449 IC50 = 135 nM T76914 C7T2IR 18009455 IC50 = 230 nM T76914 CAC32K 18009456 IC50 = 130 nM T76914 CE36ZP 18009459 IC50 = 195 nM T76914 CB3R2D 18009461 IC50 = 140 nM T76914 CIGB94 18009465 IC50 = 95 nM T76914 CMVH45 18009467 IC50 = 470 nM T76914 C5MFA8 18009473 IC50 = 230 nM T76914 C8LZI6 18009478 IC50 = 200 nM T76914 CF59QJ 18009479 IC50 = 470 nM T76914 C2CNY4 18009489 IC50 = 75 nM T76914 CLDH51 18009493 IC50 = 200 nM T76914 C76EMO 18009494 IC50 = 2790 nM T76914 C3Q4AB 18009499 IC50 = 535 nM T76914 CKI9Q7 18009506 IC50 = 245 nM T76914 C56FCT 18009507 IC50 = 150 nM T76914 CU4X1Q 18009510 IC50 > 30000 nM T76914 C8OD0P 18009511 IC50 > 30000 nM T76914 CL10UW 18009512 IC50 = 100 nM T76914 CQ0F3P 18009515 IC50 = 580 nM T76914 C41FQT 18009522 IC50 = 210 nM T76914 C1RLB8 18009528 IC50 = 120 nM T76914 C0Y9IH 18009529 IC50 = 120 nM T76914 CG8TR1 18009531 IC50 = 145 nM T76914 C4QVM5 18009534 IC50 = 8380 nM T76914 C4PS5U 18009536 IC50 = 205 nM T76914 C5H7CE 18956195 IC50 = 800 nM T76914 C43WZQ 20356975 IC50 = 5800 nM T76914 C8LAQ6 20596154 IC50 = 90 nM T76914 CU0R4A 20596162 IC50 = 420 nM T76914 CL5QI1 20596164 IC50 = 45 nM T76914 CM2P8J 20596217 IC50 > 30000 nM T76914 CAMB98 20975957 IC50 = 900 nM T76914 C7QA5W 21180801 IC50 > 100000 nM T76914 CA25KH 21404797 IC50 = 2610 nM T76914 CL0OB8 23276937 IC50 = 310 nM T76914 C91QFN 25019282 IC50 = 1410 nM T76914 CUA74K 42631042 IC50 = 15000 nM T76914 C0W2OV 42631043 IC50 > 10000 nM T76914 CUA20H 42631142 IC50 = 670 nM T76914 CX7SA6 42631143 IC50 = 890 nM T76914 CL04ZD 42631144 IC50 = 1000 nM T76914 CUW1H3 42631145 IC50 = 450 nM T76914 CSU9E8 42631146 IC50 = 12000 nM T76914 C7O1UQ 42631250 IC50 = 7000 nM T76914 CU9F7X 42631252 IC50 = 165 nM T76914 CNH6M5 42631254 IC50 = 150 nM T76914 CL45NC 42631255 IC50 = 200 nM T76914 CSIF60 42631362 IC50 = 233 nM T76914 CZ5J8O 42631363 IC50 = 1500 nM T76914 CN2IQ0 42631364 IC50 = 1000 nM T76914 CE90SQ 42631365 IC50 = 150 nM T76914 CH68ID 42631366 IC50 = 650 nM T76914 CLW7S0 42631368 IC50 = 170 nM T76914 CS7Z1Q 42631474 IC50 = 5000 nM T76914 C0OTP1 42631476 IC50 = 6000 nM T76914 CT4K6M 42631478 IC50 = 318 nM T76914 C1VS9P 42631576 IC50 = 1000 nM T76914 CT74IV 42631577 IC50 = 1000 nM T76914 C5B9LX 42631578 IC50 = 17 nM T76914 CZ1V9W 44270827 IC50 > 30000 nM T76914 CL60OE 44270838 IC50 = 325 nM T76914 CRU54T 44270847 IC50 = 10000 nM T76914 C6WOS2 44270848 IC50 > 30000 nM T76914 CW2ZN0 44270849 IC50 = 30000 nM T76914 C73SYZ 44270850 IC50 = 600 nM T76914 COZ35H 44270872 IC50 > 30000 nM T76914 CUSX95 44270881 IC50 = 690 nM T76914 CGH17I 44270891 IC50 = 780 nM T76914 C3WA7K 44270907 IC50 > 30000 nM T76914 CIX4G3 44290049 IC50 = 86 nM T76914 CO36RU 44290071 IC50 = 3200 nM T76914 C7FO3J 44298555 IC50 = 7680 nM T76914 CF84LV 44298575 IC50 > 10000 nM T76914 C79BNG 44298588 IC50 = 280 nM T76914 C49TRF 44298601 IC50 = 206 nM T76914 CBNZ03 44298603 IC50 > 10000 nM T76914 CK37YG 44298617 IC50 = 1170 nM T76914 C7ZV1G 44298618 IC50 = 817 nM T76914 CK94ZP 44298647 IC50 = 190 nM T76914 CGV9F6 44298853 IC50 > 30000 nM T76914 C5T6GQ 44298854 IC50 > 10000 nM T76914 C23EZL 44298968 IC50 = 100 nM T76914 CO4R0P 44299006 IC50 = 75 nM T76914 C2DL0U 44299007 IC50 = 279 nM T76914 CQ0S7R 44299008 IC50 = 2300 nM T76914 CZ0S6W 44299035 IC50 = 259 nM T76914 C0MQH9 44299036 IC50 = 240 nM T76914 CDZW60 44299038 IC50 = 930 nM T76914 CI3M0A 44299070 IC50 = 2620 nM T76914 C6AKB7 44299071 IC50 = 249 nM T76914 C96RUS 44299245 IC50 > 8000 nM T76914 CU04MD 44299264 IC50 > 5000 nM T76914 CFP95M 44339766 IC50 = 3900 nM T76914 CK7O4Q 44339770 IC50 = 6100 nM T76914 C8A9IX 44339771 IC50 = 5800 nM T76914 C2U6MI 44339772 IC50 = 5600 nM T76914 COH26Y 44339773 IC50 = 4000 nM T76914 CZFG53 44339790 IC50 = 10100 nM T76914 CJV4E0 44339791 IC50 = 9900 nM T76914 CH3B1G 44339837 IC50 = 9700 nM T76914 C3OBC1 44339850 IC50 = 8000 nM T76914 CR53CJ 44339937 IC50 = 3700 nM T76914 C2B1XK 44388822 IC50 = 14 nM T76914 CX04RV 44388823 IC50 = 17 nM T76914 C29CDQ 44388824 IC50 = 145 nM T76914 CRN95H 44388850 IC50 = 352 nM T76914 C9SD4N 44388851 IC50 = 19 nM T76914 C4AE7Y 44388852 IC50 = 28 nM T76914 CIQD78 44388853 IC50 = 12.3 nM T76914 CM39OU 44388873 IC50 = 29.2 nM T76914 CU3KS7 44388874 IC50 = 12 nM T76914 CA0R9F 44388875 IC50 = 21 nM T76914 CKI49B 44388876 IC50 = 48 nM T76914 CCZ9H2 44388932 IC50 = 5600 nM T76914 C9V6YM 44388933 IC50 = 1814 nM T76914 CPG79J 44388937 IC50 = 102 nM T76914 CO4G9V 44388940 IC50 = 19 nM T76914 C92VJC 44388941 IC50 = 25.5 nM T76914 C68OTU 44388942 IC50 = 11 nM T76914 CLS87F 44388957 IC50 = 143 nM T76914 CW5R7I 44388959 IC50 = 664 nM T76914 CE4F5U 44388960 IC50 = 21 nM T76914 CG5F9B 44388961 IC50 = 2000 nM T76914 CUYV21 44388976 IC50 = 380 nM T76914 CNV15W 44388977 IC50 = 26 nM T76914 C5OEG3 44388978 IC50 = 150 nM T76914 C2Z1OU 44388979 IC50 = 270 nM T76914 CD6L1X 44388992 IC50 = 74 nM T76914 CY6RN9 44388993 IC50 = 87 nM T76914 CMS7B2 44388994 IC50 = 41 nM T76914 CVPL65 44388996 IC50 = 26 nM T76914 CYV3F1 44389007 IC50 = 31 nM T76914 CMP50X 44389008 IC50 = 14 nM T76914 CE2R8P 44389009 IC50 = 34 nM T76914 CJY1M6 44389014 IC50 = 24 nM T76914 C92AQR 44389019 IC50 = 10 nM T76914 C5NYO9 44389020 IC50 = 35 nM T76914 C5XS2N 44389031 IC50 = 130 nM T76914 CA58TZ 44389032 IC50 = 200 nM T76914 CA2GE4 44389033 IC50 = 19 nM T76914 CS1OZ0 44389034 IC50 = 120 nM T76914 CRE4G2 44453927 EC50 = 1700 nM T76914 C5VFT6 44453929 EC50 = 2400 nM T76914 C7UEN0 44453949 EC50 = 2400 nM T76914 CO6X7B 44453951 EC50 = 3000 nM T76914 C4ET6C 44581197 IC50 = 2500 nM T76914 CK0MI8 44581747 IC50 = 3700 nM T76914 CRV2X0 44592608 IC50 = 7400 nM T76914 CV6M3L 44592609 IC50 = 1900 nM T76914 CFL0M1 44592610 IC50 = 4200 nM T76914 C7HTN9 44592649 IC50 = 1000 nM T76914 C6SX0U 44592650 IC50 = 1400 nM T76914 CO95DS 44592652 IC50 = 1500 nM T76914 CC8AB9 44592686 IC50 < 3000 nM T76914 CVA0U7 44592687 IC50 = 1500 nM T76914 CW8M0G 44592720 IC50 = 710 nM T76914 CGT69F 44592757 IC50 > 10000 nM T76914 C9PC8V 44592758 IC50 = 6100 nM T76914 CZ9M2W 44592759 IC50 = 3600 nM T76914 CN1PC9 44592783 IC50 = 13000 nM T76914 C3ESW7 44592784 IC50 = 4000 nM T76914 C46XRM 44592785 IC50 = 3400 nM T76914 C73DZF 44593040 IC50 < 2000 nM T76914 CUFK03 45271233 IC50 = 520 nM T76914 C76ULT 50908597 IC50 = 930 nM T76914 C10CAI 50908735 IC50 = 350 nM T76914 CNP3Q6 50908736 IC50 = 250 nM T76914 CWZ65U 50908897 IC50 = 550 nM T76914 C0N7SB 50908898 IC50 = 700 nM T76914 C6ICT2 50908899 IC50 = 370 nM T76914 C5OG2J 50908900 IC50 = 820 nM T76914 C7EB3O 52941155 IC50 = 360 nM T76914 CV4JG5 52941196 IC50 = 17500 nM T76914 CZ92PU 52941197 IC50 = 37400 nM T76914 CVB2S3 52941198 IC50 = 330 nM T76914 C5GD7U 52941223 IC50 = 670 nM T76914 CZ2YP1 52941279 IC50 = 470 nM T76914 CTMB85 52941304 IC50 = 4700 nM T76914 CU23TL 52941375 IC50 = 1180 nM T76914 CH29GZ 52941394 IC50 = 820 nM T76914 CG2TW3 52941465 IC50 = 230 nM T76914 CDB2H0 52941558 IC50 = 1390 nM T76914 CYU9F4 52941559 IC50 = 350 nM T76914 CL6P5Z 52941606 IC50 = 14700 nM T76914 CS1C3E 52941613 IC50 = 5900 nM T76914 C40OFP 52941700 IC50 = 550 nM T76914 CUY46W 52942353 IC50 = 11200 nM T76914 CBJ50X 52942519 IC50 > 50000 nM T76914 C0SR8T 52942627 IC50 = 2950 nM T76914 CSX39T 52942698 IC50 = 5160 nM T76914 CW1N6Z 52942757 IC50 = 15300 nM T76914 C2CZX9 52942766 IC50 = 1550 nM T76914 CH7KN9 52942767 IC50 = 470 nM T76914 C3YM0N 52942845 IC50 > 50000 nM T76914 CNLZ56 52942888 IC50 = 2670 nM T76914 C5KB1P 52943563 IC50 = 2870 nM T76914 CBE14N 52943618 IC50 > 50000 nM T76914 C4TX1V 52943646 IC50 = 1050 nM T76914 C3MIL9 52943647 IC50 = 1300 nM T76914 CFD46Z 52943648 IC50 = 160 nM T76914 C84XGP 52943813 IC50 = 1150 nM T76914 CW9DO1 52943894 IC50 = 200 nM T76914 C03IQO 52943946 IC50 = 2660 nM T76914 CF4YT9 52943984 IC50 = 730 nM T76914 C9VHK1 52943985 IC50 = 1510 nM T76914 CB96VD 52944057 IC50 = 1350 nM T76914 CYF0S3 52944791 IC50 = 910 nM T76914 C5CN7Y 52944792 IC50 = 640 nM T76914 CA0QV6 52944811 IC50 = 3490 nM T76914 CIW8Q2 52944838 IC50 = 2560 nM T76914 CQ02KD 52944866 IC50 = 3400 nM T76914 CL23DS 52944926 IC50 = 700 nM T76914 C1PAQ4 52944957 IC50 = 200 nM T76914 CN35LH 52944958 IC50 = 150 nM T76914 C9PX5E 52944999 IC50 = 300 nM T76914 C3DYJ5 52945000 IC50 = 540 nM T76914 C0O4CT 52945029 IC50 = 550 nM T76914 C6E7QV 52945057 IC50 = 4810 nM T76914 C0AFU8 52945163 IC50 = 140 nM T76914 CH8G2D 52945193 IC50 = 2430 nM T76914 C4X9LB 52945279 IC50 > 50000 nM T76914 CZ50SQ 52946006 IC50 = 630 nM T76914 C97ALI 52946105 IC50 > 50000 nM T76914 CIN90C 52946106 IC50 > 50000 nM T76914 CZ3P4V 52946157 IC50 = 560 nM T76914 CE6AT5 52946186 IC50 = 700 nM T76914 CGU07R 52946227 IC50 = 31600 nM T76914 C5P6LQ 52946269 IC50 > 50000 nM T76914 CV31NF 52946270 IC50 = 150 nM T76914 CIV24B 52946310 IC50 = 13100 nM T76914 CX6EF7 52946321 IC50 = 16400 nM T76914 CX8C5G 52946322 IC50 > 50000 nM T76914 CD9S1F 52946334 IC50 = 7200 nM T76914 C4ED8W 52946335 IC50 = 530 nM T76914 C8R1ZO 52946384 IC50 = 200 nM T76914 C6YG9U 52946418 IC50 = 1080 nM T76914 CEYS37 52946495 IC50 = 15500 nM T76914 CJ7AY2 52946550 IC50 = 10100 nM T76914 CXI3M6 52947252 IC50 > 50000 nM T76914 C9WRK4 52947357 IC50 = 12000 nM T76914 CYS6C8 52947504 IC50 > 15800 nM T76914 CRT45X 52947623 IC50 = 2390 nM T76914 CZ3HN6 52947639 IC50 = 310 nM T76914 CAE61M 52948439 IC50 = 850 nM T76914 CR8H2T 52948440 IC50 > 50000 nM T76914 C28QEH 52948441 IC50 = 390 nM T76914 CJ1RH6 52948489 IC50 = 840 nM T76914 CU89SW 52948510 IC50 = 1070 nM T76914 CWA9F3 52948583 IC50 = 340 nM T76914 CMG1Z5 52948605 IC50 = 1260 nM T76914 CLO5M6 52948637 IC50 = 6750 nM T76914 CHR08Q 52948676 IC50 = 16300 nM T76914 C0LCS3 52948698 IC50 = 280 nM T76914 CZT6C4 52948768 IC50 > 50000 nM T76914 CO58DG 52948836 IC50 = 3590 nM T76914 C4IL2V 52948983 IC50 = 750 nM T76914 CAB7U5 52948996 IC50 = 90 nM T76914 CJ95MD 52949687 IC50 = 500 nM T76914 C5PO9R 52949704 IC50 > 50000 nM T76914 C3DSB1 52949759 IC50 = 440 nM T76914 CG9MB0 52949844 IC50 = 530 nM T76914 CVA21P 52949880 IC50 = 9790 nM T76914 CF6U3A 52949881 IC50 > 50000 nM T76914 C9LSE2 52949905 IC50 = 2350 nM T76914 C46JBA 52949924 IC50 = 3080 nM T76914 C43YBI 52949966 IC50 = 80 nM T76914 C1FOZ0 52949971 IC50 = 320 nM T76914 C4G7ZT 52950023 IC50 = 880 nM T76914 C8J1GU 52950034 IC50 = 2750 nM T76914 COC51A 58282550 IC50 = 75000 nM T76914 CQZH53 71452336 IC50 = 4200 nM T76914 C74LEQ 71454124 IC50 = 230000 nM T76914 C5YQ1P 71455850 IC50 = 2520 nM T76914 C0LFZ2 71455851 IC50 = 25000 nM T76914 CHU57F 71457657 IC50 > 100000 nM T76914 C4QTY2 71459549 IC50 > 100000 nM T76914 C9OB0I 71463015 IC50 = 750 nM T76914 CM4H3O 71463016 IC50 > 100000 nM T76914 CQSZ72 90675942 IC50 = 21000 nM T76914 CTBD74 90675943 IC50 = 14000 nM T76914 CM12LR 102597975 IC50 = 1400 nM T76914 CQJ49Y 122187245 IC50 = 0.375 nM T76914 CSW57U 122187246 IC50 = 0.111 nM T76914 C98BUE 122187247 IC50 = 0.042 nM T76914 CVT7A6 122187248 IC50 = 0.046 nM T76914 CI9ZH1 122187249 IC50 = 0.07 nM T76914 CHJ75V 122187250 IC50 = 0.201 nM T76914 C20TPX 122187251 IC50 = 0.034 nM T76914 CQ17ZP 122187252 IC50 = 0.045 nM T76914 C2XUA5 122187253 IC50 = 0.159 nM T76914 CQTJ57 122187272 IC50 = 0.11 nM T76914 CX2YG6 122187273 IC50 = 0.216 nM T76914 C4CLN5 122187274 IC50 > 3.333 nM T76914 CF5M8V 122187275 IC50 = 18.5 nM T76914 C24MEW 122187276 IC50 > 3.333 nM T76914 CI7VL5 122187277 IC50 > 3.333 nM T76914 COX2P3 122187278 IC50 = 1.11 nM T76914 CY9RL0 122187279 IC50 = 0.245 nM T76914 CT5B4D 122187280 IC50 = 0.202 nM T76914 C42SZA 122187281 IC50 = 8.16 nM T76914 C6S3XG 122187282 IC50 = 0.143 nM T76914 C0YG3Z 122187283 IC50 = 0.043 nM T76914 C1F5PE 122187284 IC50 = 0.234 nM T76914 C26VHJ 122187285 IC50 = 0.176 nM T76914 C24JCI 122187286 IC50 = 0.073 nM T76914 CW4SU9 122187287 IC50 = 0.074 nM T76914 CT0GS6 122187288 IC50 = 0.098 nM T76914 CCO3Y2 122187289 IC50 > 3.333 nM T76914 C1ENW4 122187290 IC50 = 0.215 nM T76914 CFH36G 122187291 IC50 = 6.56 nM T76914 C3CY5N 122187292 IC50 = 0.253 nM T76914 CY69QI 122187293 IC50 = 0.083 nM T76914 C05WQZ 122187294 IC50 = 0.072 nM T76914 C1LW9V 122187295 IC50 = 0.398 nM T76914 CBMT85 122187296 IC50 = 0.205 nM T76914 C8AKN9 122187297 IC50 = 0.143 nM T76914 CDM71F 122187298 IC50 = 0.166 nM T76914 CCM08N 122187299 IC50 = 0.056 nM T76914 C7V2TW 122187300 IC50 = 0.095 nM T76914 C81QSJ 122187301 IC50 = 25.3 nM T76914 C1IPG9 122187302 IC50 = 3.08 nM T76914 C0RE2W 122187303 IC50 > 3.333 nM T76914 C9JDM3 122187304 IC50 > 3.333 nM T76914 C5QXR6 122187305 IC50 = 0.094 nM T76914 C50RMQ 122187306 IC50 = 0.107 nM T76914 C5Z9PU 122187307 IC50 = 0.158 nM T76914 CT0V4W 122187308 IC50 = 13 nM T76914 CX06CZ 122187309 IC50 = 0.038 nM T76914 CK9T7F 122187310 IC50 > 3.333 nM T76914 CC2LE0 122187311 IC50 = 0.089 nM T76914 CS34VD 122187312 IC50 = 0.357 nM T76914 CIU9T5 122187313 IC50 = 0.154 nM T76914 CS8QW7 122187314 IC50 = 0.023 nM T76914 CID97N 122187315 IC50 > 3.333 nM T76914 CZ08GP 122187316 IC50 = 0.117 nM T76914 C0P6IC 122187317 IC50 = 0.561 nM T76914 CY7M0F 122187318 IC50 = 0.083 nM T76914 CQZK10 122187319 IC50 = 0.052 nM T76914 C62FDT 122187320 IC50 = 0.095 nM T76914 C3QZY1 122187321 IC50 = 0.154 nM T76914 C8B4YL 122187322 IC50 = 0.073 nM T76914 CWV12K 122187323 IC50 = 0.991 nM T76914 CWVP15 122187324 IC50 = 0.108 nM T76914 CEW35A 122187325 IC50 = 0.041 nM T76914 CP43GQ 122187326 IC50 = 0.108 nM T76914 CH46BC 122187327 IC50 = 0.798 nM T76914 C6KW2B 122187328 IC50 = 0.108 nM T76914 C87MGD 122187329 IC50 = 0.1 nM T76914 C0U9QN 122187330 IC50 = 0.122 nM T76914 CH4G1L 122187331 IC50 = 3.49 nM T76914 C4ZR9M 122187332 IC50 = 0.041 nM T76914 CM8A1Y 122187333 IC50 = 1.417 nM T76914 CU3IE9 122187334 IC50 = 0.122 nM T76914 CYN12K 122187335 IC50 = 0.067 nM T76914 CDE52G 122187336 IC50 = 0.138 nM T76914 CZH25J 122187337 IC50 = 0.082 nM T76914 CQP1R4 122187338 IC50 = 0.223 nM T76914 C3QS0A 122187339 IC50 = 0.138 nM T76914 CAFO71 122187340 IC50 = 0.04 nM T76914 CNYJ15 122187341 IC50 = 0.13 nM T76914 CY62QW 122187342 IC50 = 0.153 nM T76914 CCV2G0 122187343 IC50 = 0.305 nM T76914 C0Z8JH 122187344 IC50 = 0.037 nM T76914 CVT8Z7 122187345 IC50 = 3.763 nM T76914 C2YI7W 122187346 IC50 = 0.031 nM T76914 CO7MU2 122187445 IC50 = 0.431 nM T76914 C8QN9Z 122187446 IC50 = 0.795 nM T76914 C09YUX 122187447 IC50 = 0.041 nM T76914 C8I6TF 122187448 IC50 = 0.054 nM T76914 CR68ZK 122187449 IC50 = 0.032 nM T76914 CTY96B 122187450 IC50 = 0.24 nM T76914 C4WG0M 122187451 IC50 = 0.251 nM T76914 CLS4H7 122187452 IC50 = 0.227 nM T76914 CM23CQ 122187453 IC50 = 0.456 nM T76914 CJF8X1 122187454 IC50 = 0.261 nM T76914 C54PSK 122187455 IC50 = 0.045 nM T76914 CGS5Q1 122187456 IC50 = 0.641 nM T76914 CW0MH4 122187457 IC50 = 0.135 nM T76914 CXAV52 122187458 IC50 = 8.01 nM T76914 C3D8EQ 122187459 IC50 = 2.88 nM T76914 CBUT59 122187460 IC50 = 0.173 nM T76914 C1XL3M 122187461 IC50 = 0.039 nM T76914 CBS95M 122187462 IC50 = 0.059 nM T76914 CY79JC 122187463 IC50 = 0.083 nM T76914 CAY0P4 122187464 IC50 = 0.223 nM T76914 CRQ98D 122187465 IC50 = 0.223 nM T76914 CXP98T 122187466 IC50 = 0.318 nM T76914 C5TJU8 122187467 IC50 > 3.333 nM T76914 CP7C2I 122187468 IC50 = 0.86 nM T76914 CKC0L8 122187469 IC50 > 3.333 nM T76914 CV3T2C 122187470 IC50 = 0.368 nM T76914 CN5OQ2 122187471 IC50 = 0.205 nM T76914 CI0J4A 122187472 IC50 = 0.927 nM T76914 CM14KC 122187473 IC50 = 0.235 nM T76914 COFI26 122187474 IC50 = 0.039 nM T76914 CTXG58 122187475 IC50 = 0.073 nM T76914 CZWG59 122187476 IC50 = 9.55 nM T76914 C1TVY5 122187477 IC50 = 0.153 nM T76914 CS6FK8 122187478 IC50 > 100 nM T76914 CJC21F 122187479 IC50 = 0.853 nM T76914 C3ZE4Y 122187480 IC50 > 100 nM T76914 CS0U8H 122187481 IC50 > 3.333 nM T76914 CY0NV5 122187482 IC50 = 0.061 nM T76914 C8SHE5 122187483 IC50 = 0.207 nM T76914 CHYI14 122187484 IC50 = 0.223 nM T76914 CEH14V 122187485 IC50 > 3.333 nM T76914 CG98KU 122187486 IC50 = 0.082 nM T76914 C3P8WN 122187487 IC50 = 0.032 nM T76914 C9MJ2K 122187488 IC50 = 0.182 nM T76914 C7J0YH 122187489 IC50 = 0.077 nM T76914 C4NYT7 122187490 IC50 = 0.151 nM T76914 CMT25I 122187491 IC50 = 0.029 nM T76914 CQEV80 122187492 IC50 = 0.031 nM T76914 CY07HP 122187493 IC50 = 16.9 nM T76914 CD0EU3 122187494 IC50 = 0.074 nM T76914 CQZ0R1 122187495 IC50 = 1.308 nM T76914 CZU4N2 122187496 IC50 = 0.072 nM T76914 CITK91 122187497 IC50 = 0.056 nM T76914 C69JKA 122187498 IC50 = 0.023 nM T76914 C6R5CY 122187499 IC50 = 0.983 nM T76914 CM87YE 122187500 IC50 = 0.152 nM T76914 CP4GJ7 122187501 IC50 = 0.352 nM T76914 CB14ES 122187502 IC50 = 0.047 nM T76914 CEGB98 122187503 IC50 = 0.267 nM T76914 C1GY9X 135402606 IC50 > 50000 nM T76914 CYOD40 145964126 IC50 > 30000 nM T76914 CW9P6A 145964460 IC50 = 17000 nM T76914 CQR49Z 145965116 IC50 = 25000 nM T76914 CF6C3J 145966416 IC50 > 30000 nM T76914 CFM10D 145967283 IC50 > 30000 nM T76914 CR6L2G 145967358 IC50 = 9000 nM T76914 CI96RT 145970087 IC50 > 30000 nM T76914 CI6MO5 145973473 IC50 > 30000 nM T76914 CFG05L 145975803 IC50 > 30000 nM T76914 CN03BP 145976644 IC50 > 30000 nM T76914 CHXE25 145978207 IC50 = 25000 nM T76914 D04UVC 44270882 IC50 = 150 nM T76914 D05RLR 656734 IC50 = 5000 nM T76914 D07VWP 656730 IC50 = 2300 nM T76914 D08BMM 6312649 IC50 = 4700 nM T76914 D0A4LH 602095 IC50 = 5800 nM T76914 D0CI6E 44389018 IC50 = 100 nM T76914 D0E9MC 656767 IC50 = 200 nM T76914 D0H1EI 6603977 IC50 = 724 nM T76914 D0L0FC 44298928 IC50 = 164 nM T76914 D0R9CF 11302540 IC50 = 2 nM T76914 D0S8CL 10433084 IC50 = 828 nM T92963 C0EDH1 44301581 Ki = 62 nM T92963 C4T0MB 44301645 Ki = 680 nM T92963 C8M2XU 44301646 Ki = 0.3 nM T92963 C9AME2 44301661 Ki = 1.64 nM T92963 CZ4Y6B 44301714 Ki = 0.48 nM T92963 CRQ1L0 44301718 Ki = 0.49 nM T92963 C9SZ3D 44301732 Ki = 0.4 nM T92963 C02LJW 44301739 Ki = 65 nM T92963 CE0AU3 44301746 Ki = 2600 nM T92963 CDCM97 44301748 Ki = 2900 nM T92963 C5O3NG 44301749 Ki = 539 nM T92963 CGO6W5 44301973 Ki = 87 nM T92963 CDV2Z1 131717293 IC50 = 1.5 nM T92963 CE1IC8 137636347 IC50 = 0.079 nM T92963 CJX30M 137636606 IC50 = 0.087 nM T92963 C3CA5Q 137636877 IC50 = 0.93 nM T92963 COA5V7 137637572 IC50 = 0.054 nM T92963 CLB82Z 137638007 IC50 = 0.12 nM T92963 C19FLA 137639109 IC50 = 0.36 nM T92963 CKC79W 137640954 IC50 = 35 nM T92963 CF8TO7 137642743 IC50 = 0.52 nM T92963 CQEP84 137642780 IC50 = 0.14 nM T92963 C4DHJ5 137643645 IC50 = 11 nM T92963 CK6U0S 137645853 IC50 = 0.13 nM T92963 CHW8M5 137646261 IC50 = 0.65 nM T92963 CAZC92 137646317 IC50 = 0.19 nM T92963 CJ2PC6 137648579 IC50 = 0.3 nM T92963 C4RHT7 137649996 IC50 = 7.8 nM T92963 CFV35E 137649998 IC50 = 0.12 nM T92963 CWG42U 137651404 IC50 = 15 nM T92963 CVY34O 137652046 IC50 = 1.2 nM T92963 C47ZKI 137652546 IC50 = 13 nM T92963 C49CYT 137654685 IC50 = 22 nM T92963 CX6M5O 137656853 IC50 = 13 nM T92963 CEC4S2 137657880 IC50 = 0.51 nM T92963 CWH19J 137659661 IC50 = 54 nM T92963 CY89PF 137660705 IC50 = 0.099 nM T92963 CVX3W8 137662168 IC50 = 0.058 nM T04773 CF1AK9 5346177 Ki > 10000 nM T04773 C5YHI6 5346361 Ki > 10000 nM T04773 C3HZM9 5356341 Ki = 625 nM T04773 C4A1LY 5708902 Ki > 10000 nM T04773 CL45FU 5708903 Ki = 53 nM T04773 C5GX3C 5951757 Ki = 1380 nM T04773 CZ4YD0 6082907 Ki > 10000 nM T04773 C0ZV9S 6123890 Ki > 10000 nM T04773 CY5W1M 6123893 Ki = 285 nM T04773 CE7L8T 6171844 Ki = 1780 nM T04773 CH7B3C 6179219 Ki > 10000 nM T04773 C3EK9R 6266712 Ki = 44 nM T04773 CL0Y1K 7528837 Ki > 10000 nM T04773 C9NZI1 8828521 Ki = 25 nM T04773 C8XRJ4 8856159 Ki = 430 nM T04773 C9K0GV 8856731 Ki = 714 nM T04773 CW1A4Y 8858264 Ki = 53 nM T04773 CML31K 8858318 Ki = 48 nM T04773 C4N5YT 10494611 Ki > 10000 nM T04773 CK5N1Y 14977361 Ki = 350 nM T04773 C3N7PW 15354441 Ki = 107 nM T04773 CQ23RP 15354445 Ki > 10000 nM T04773 CLQ6S3 21436904 Ki > 10000 nM T04773 CX5K8H 25266037 Ki = 1070 nM T04773 CWJ59X 36074997 Ki = 107 nM T04773 CDWK49 134180849 Ki = 107 nM T04773 CE30UP 137287575 Ki = 267 nM T04773 CUX13T 145949318 Ki > 10000 nM T04773 C7JEN4 145949325 Ki > 10000 nM T04773 CTE06C 145949383 Ki = 357 nM T04773 CI9RY1 145949748 Ki > 5000 nM T04773 C0LAI8 145949999 Ki = 357 nM T04773 C3F8DV 145951494 Ki = 496 nM T04773 C5CU2V 145951688 Ki > 10000 nM T04773 CBC85F 145952108 Ki > 10000 nM T04773 CNRT31 145952390 Ki = 71 nM T04773 C6DHL3 145955526 Ki = 107 nM T04773 C6NB3E 145955922 Ki = 1071 nM T04773 C10OXY 145956615 Ki = 475 nM T04773 C8YCV2 145956775 Ki = 357 nM T04773 CHS5V8 145957162 Ki = 203 nM T04773 C74VSG 145957751 Ki = 107 nM T04773 CP4A5X 145959486 Ki > 10000 nM T04773 C8Q1NH 145959772 Ki = 1680 nM T04773 CG31CE 145960042 Ki > 10000 nM T04773 CZT34E 145971277 Ki = 5350 nM T04773 CQG27P 145972252 Ki > 10000 nM T79232 D04JEE 4946 EC50 > 5011.87 nM T79232 D08FJL 16681432 EC50 = 2.3 nM T79232 D0D8XY 5311010 Ki = 0.15 nM T79232 D0F4NS 119369 Ki = 195 nM T79232 D0M3FJ 439302 EC50 = 0.18 nM T79232 D0N4OW 644077 EC50 = 0.004 nM T79232 D0U7SH 5311065 Ki = 62.4 nM T79232 D0VU2X 151171 Ki = 0.43 nM T79232 D04QZI 11340891 Ki > 12000 nM T79232 D07EEN 172997 Ki = 44 nM T79232 D09WYL 11634973 Ki > 6309.57 nM T79232 D0F4VW 44428550 Ki = 0.3 nM T79232 D0G2XE 6918468 IC50 = 740 nM T79232 D0L6XQ 11157078 IC50 = 38 nM T79232 D0L9NX 158348 Ki = 304 nM T79232 D0LI1C 44469321 IC50 > 10000 nM T79232 D0PB0D 11686429 Ki = 0.66 nM T79232 D0S3YN 53330936 EC50 = 2.399 nM T79232 D0SY9B 9895468 Ki = 22 nM T79232 D03RYS 5311500 Ki = 344 nM T79232 D08ORO 114904 Ki = 350 nM T79232 D08PAC 6918320 Ki < 1995.26 nM T79232 D0A1KU 11683187 Ki = 1120 nM T79232 D0AV0O 3038506 Ki = 819 nM T79232 D0I8ZZ 60943 Ki = 0.19 nM T79232 D0Q8RX 9872389 Ki = 180 nM T79232 C0R7SI 449224 EC50 = 3.2 nM T79232 CZN6S9 743974 IC50 > 50118.72 nM T79232 CI82HM 999998 Ki = 325 nM T79232 C5F1ST 1103817 Ki = 1410 nM T79232 CESI60 1134581 Ki = 300 nM T79232 C0WY8H 1134627 Ki = 70 nM T79232 CIAB57 1135733 Ki = 115 nM T79232 CZN48Y 1153909 Ki > 10000 nM T79232 C2HKQ3 1153925 Ki > 10000 nM T79232 C1UAI6 1368921 Ki > 10000 nM T79232 C0AB3Y 3601935 EC50 = 0.1259 nM T79232 CX05TJ 4391207 IC50 = 200 nM T79232 CQZF41 5002508 Ki > 10000 nM T79232 C1C3LR 5014150 EC50 = 0.1585 nM T79232 C7AD6Y 5034737 Ki = 120 nM T79232 CQB93O 5306925 Ki = 556 nM T79232 CM6VF8 6734379 IC50 = 2010 nM T79232 C93WRU 9690136 Ki = 170 nM T79232 C5E3XU 9799174 IC50 = 3 nM T79232 CC07MW 9807249 Ki = 24 nM T79232 CC24MQ 9807250 Ki = 640 nM T79232 CO3SD6 9811830 EC50 = 0.2692 nM T79232 CO9VA3 9820671 IC50 > 1000 nM T79232 CML46C 9824954 IC50 = 5954 nM T79232 C57WZH 9826033 IC50 = 3100 nM T79232 CS8Q6R 9826254 IC50 = 15 nM T79232 CW8ZA7 9828129 IC50 = 1140 nM T79232 C6OV5R 9829108 IC50 = 126 nM T79232 C6RU1S 9833460 Ki = 0.39 nM T79232 CQYU70 9849525 Ki = 49 nM T79232 CA7RO2 9871426 IC50 = 729 nM T79232 C7SMT0 9908904 IC50 > 1000 nM T79232 CDFI62 9915472 IC50 = 24 nM T79232 CRM93H 9931699 IC50 = 1783 nM T79232 C8IW4K 9935206 IC50 = 0.5 nM T79232 C1C6HA 9937535 IC50 = 4 nM T79232 COUA25 9938406 Ki = 740 nM T79232 CNJ81W 9959174 Ki = 26 nM T79232 CIE8X5 9981665 Ki = 1600 nM T79232 C9J4MZ 10003306 IC50 = 20 nM T79232 CT7SZ8 10119966 Ki = 40 nM T79232 C1C4SX 10142915 Ki = 4.5 nM T79232 C98HVI 10144208 Ki = 8.09 nM T79232 C68ZRW 10156521 IC50 = 88 nM T79232 CL71MC 10164478 Ki = 1.04 nM T79232 C2NEU9 10165683 Ki = 13.2 nM T79232 C7VW8K 10187283 Ki = 3.03 nM T79232 CV7A0N 10206901 Ki = 13.9 nM T79232 CPEN43 10208363 Ki = 570 nM T79232 CPE3F8 10208389 Ki = 1.46 nM T79232 CV2Z3J 10278394 Ki = 4.09 nM T79232 CH2XI7 10279928 IC50 ~ 100 nM T79232 C4LU8J 10303620 Ki = 1.05 nM T79232 C52SOK 10304617 Ki = 1.01 nM T79232 C15PBH 10318802 IC50 = 18 nM T79232 CF6A5Y 10322392 IC50 = 8 nM T79232 CW50TU 10345610 IC50 = 4.8 nM T79232 C9M0XS 10359487 IC50 = 117 nM T79232 CE0PB5 10383074 IC50 = 83 nM T79232 C06SVZ 10392505 IC50 = 4 nM T79232 CTWG68 10411308 Ki = 2.74 nM T79232 CKD75B 10414302 Ki = 84 nM T79232 C1OIW6 10416272 Ki = 1258.93 nM T79232 C8DWH6 10456892 IC50 = 1.3 nM T79232 C5JSO3 10459252 IC50 = 370 nM T79232 C1Z3WY 10461417 IC50 = 4 nM T79232 CTSQ23 10474163 IC50 = 29 nM T79232 CR6VX2 10483105 Ki = 620 nM T79232 CY58RQ 10503858 IC50 = 120 nM T79232 C2Z7RB 10587836 Ki = 734 nM T79232 C5NIU8 10648029 IC50 = 430 nM T79232 CLXT94 10672170 IC50 = 540 nM T79232 C8VB3L 10673295 IC50 = 640 nM T79232 CZKU73 10673699 IC50 = 4400 nM T79232 CYE0I7 10696913 IC50 = 32 nM T79232 CCU35N 10715974 Ki = 1.58 nM T79232 CH84ZE 10719289 IC50 = 25 nM T79232 CR8QV4 10742418 IC50 = 59 nM T79232 CL1N4A 10743786 IC50 = 37 nM T79232 CU4EL3 10766720 IC50 = 15 nM T79232 C4GTY9 10814200 IC50 = 340 nM T79232 C2TL5U 10837633 IC50 = 6.3 nM T79232 C3U6QA 10863737 Ki = 9.06 nM T79232 CQJ52W 10873853 Ki = 55.5 nM T79232 C1WD7P 10907482 Ki = 9.16 nM T79232 CT79NZ 10927276 IC50 = 5160 nM T79232 CI8AQ1 10929819 Ki = 39.4 nM T79232 CM0OS2 10939174 IC50 = 6650 nM T79232 CQ0JE5 10984025 Ki = 214 nM T79232 CGK39X 10984026 Ki > 10000 nM T79232 CJC9K4 11005810 IC50 = 3650 nM T79232 CBOS05 11016093 Ki = 2.12 nM T79232 CFJG64 11059058 IC50 = 2220 nM T79232 CFL2P5 11092056 Ki = 29.1 nM T79232 CDF9W0 11144861 Ki = 7.84 nM T79232 C0FJM7 11194023 Ki = 36.3 nM T79232 C6D3UR 11237434 IC50 = 6.7 nM T79232 C2PE4M 11238362 IC50 = 8 nM T79232 CO3A5Z 11240155 Ki = 19.7 nM T79232 CC0KT1 11251777 Ki = 36.9 nM T79232 CUED54 11257380 Ki = 388 nM T79232 CU1E4A 11261339 IC50 = 19 nM T79232 C5OTG4 11274745 Ki = 436 nM T79232 C45MWC 11278622 IC50 = 345 nM T79232 CG10YR 11282041 IC50 = 7000 nM T79232 C9T8BV 11286254 Ki = 75 nM T79232 CB6TF8 11297732 Ki = 80 nM T79232 C2TC8K 11326488 IC50 = 110 nM T79232 C2RA0J 11337030 IC50 = 133 nM T79232 CYJ23D 11384094 Ki = 132 nM T79232 CPND10 11389106 Ki = 13 nM T79232 CEM1X7 11400547 Ki = 48.2 nM T79232 CG0Q5O 11432362 IC50 = 13 nM T79232 CHJ7E2 11451056 IC50 = 9 nM T79232 CPTM67 11461755 IC50 = 71 nM T79232 CR4N5I 11465834 Ki = 630.96 nM T79232 CM83DS 11468862 Ki = 463 nM T79232 CLQ3N9 11473073 IC50 = 199 nM T79232 C37TNB 11475469 Ki = 4300 nM T79232 C9SY7Q 11486351 Ki = 1700 nM T79232 COC7Q9 11488952 Ki < 6309.57 nM T79232 CR5SH4 11502419 Ki = 24.4 nM T79232 CGU9K0 11513323 Ki = 1.49 nM T79232 CFA81S 11519251 Ki = 1800 nM T79232 C5PU0J 11538526 Ki = 111 nM T79232 CQ96XZ 11569194 Ki > 6309.57 nM T79232 C60DKW 11569672 Ki < 39810.72 nM T79232 CM15EB 11574636 Ki = 2400 nM T79232 CG7CL9 11578939 EC50 = 0.38 nM T79232 CP0U2Q 11619807 Ki = 1860 nM T79232 CD2NZ0 11620428 Ki = 1600 nM T79232 CFPR21 11625088 Ki = 21.6 nM T79232 C8D5PW 11626867 Ki > 10000 nM T79232 C60ODW 11641980 Ki > 10000 nM T79232 CQ4SX5 11667812 Ki = 608 nM T79232 CY0HE4 11677610 IC50 > 100000 nM T79232 CT41LU 11692335 Ki = 1600 nM T79232 CKF35C 11700583 Ki = 5.84 nM T79232 C0GD8A 11740204 IC50 = 17 nM T79232 CIC93G 11740743 Ki = 8.1 nM T79232 C91CIO 11815584 Ki = 1.5 nM T79232 CCQ01Y 11848692 Ki = 732 nM T79232 C8GC2P 11854507 IC50 > 100000 nM T79232 CIZ74V 11961325 IC50 = 4480 nM T79232 C2E7DV 11993729 Ki = 1 nM T79232 CIU3X9 13145539 Ki = 3.4 nM T79232 C4CTD2 14257660 EC50 = 0.69 nM T79232 C2SB0G 14306032 IC50 = 45 nM T79232 CH8F9Q 14306034 IC50 > 5000 nM T79232 CQ93UO 14306046 IC50 = 61000 nM T79232 C1E4BW 15298022 IC50 = 13 nM T79232 CEI74X 15307998 IC50 = 36 nM T79232 CIDT94 15307999 IC50 = 43 nM T79232 CMP0I2 15308000 IC50 = 8.5 nM T79232 C06DHE 15416417 Ki = 1.85 nM T79232 CU3M1I 15416418 Ki = 1.03 nM T79232 CTEW91 15951937 Ki = 4 nM T79232 CDU6Z8 15952030 Ki = 32 nM T79232 CXRY43 15952129 Ki = 16 nM T79232 C1SKJ3 15953022 Ki = 2 nM T79232 CR2B0I 15976308 Ki = 1.89 nM T79232 CHU5E4 16051933 Ki = 3.8 nM T79232 CQM10O 16059348 Ki = 8 nM T79232 C7T2WZ 16062053 Ki = 525 nM T79232 CSRL29 16063234 Ki = 118 nM T79232 CY6EU0 17757748 Ki = 32 nM T79232 CNL0G2 17989455 IC50 = 20 nM T79232 C8CY9A 19607875 Ki = 910 nM T79232 CGDY68 19608069 Ki = 68 nM T79232 CGC20J 19699093 IC50 = 240 nM T79232 CY89CI 19699133 IC50 = 4100 nM T79232 C6TKQ8 20825285 IC50 = 35 nM T79232 C60ALS 21064021 IC50 = 5380 nM T79232 CEH7B3 21064040 IC50 = 135 nM T79232 CCD46Q 21467141 IC50 = 86 nM T79232 CUV4H1 21925546 IC50 = 345 nM T79232 C6CT4M 21925559 IC50 = 904 nM T79232 C12QOU 21925586 IC50 = 272 nM T79232 CESD54 21925639 IC50 = 17 nM T79232 C1E7AB 22017577 IC50 = 25 nM T79232 C4Y6GR 22017582 IC50 = 2460 nM T79232 CMAS73 22017591 IC50 = 20 nM T79232 CG7JW4 22162609 EC50 > 100 nM T79232 C59LDI 22405322 IC50 = 12 nM T79232 C64FDO 22405324 IC50 = 21 nM T79232 CUD2I8 22405325 IC50 = 63 nM T79232 CX89MH 22405326 IC50 = 280 nM T79232 CGD49J 22405327 IC50 = 64 nM T79232 CW7O1M 22405331 IC50 = 85 nM T79232 C2DXS5 22861321 IC50 = 13 nM T79232 CE4Z6R 23598556 IC50 = 10 nM T79232 CEOZ91 23598560 IC50 = 26 nM T79232 C71XOU 23598595 IC50 = 20 nM T79232 CBRI52 23598597 IC50 = 11600 nM T79232 CJ8Z6N 23598598 IC50 = 10 nM T79232 CM1F7K 23598600 IC50 = 19 nM T79232 CP8GK0 23598619 IC50 = 15 nM T79232 C4G8ZR 23598638 IC50 = 100 nM T79232 CPZE93 23598641 IC50 = 9 nM T79232 CP64WA 23598642 IC50 = 630 nM T79232 CW0C3M 24894462 Ki = 10.5 nM T79232 C4T5HX 24894463 Ki = 30 nM T79232 CTV17B 24896178 Ki = 1.17 nM T79232 CBT8A3 24958835 Ki = 81 nM T79232 CG2B5X 24997177 Ki = 5 nM T79232 CC0X3Y 25001616 Ki = 39 nM T79232 CN5HE0 25001929 Ki = 9 nM T79232 C7NJ1B 25109291 Ki = 2.4 nM T79232 CG20SB 25132666 IC50 = 63 nM T79232 C7C1TG 25132999 IC50 = 320 nM T79232 CWSF74 25133000 IC50 = 27 nM T79232 C3Q0AD 25133001 IC50 = 95 nM T79232 COC73W 25212177 Ki = 63.1 nM T79232 CCX14Y 26434734 Ki = 82 nM T79232 CY67HA 42611262 Ki = 12.59 nM T79232 CAM63X 42618195 IC50 > 1000 nM T79232 C8K4UF 42618197 IC50 > 1000 nM T79232 CS04KE 42629368 Ki = 6300 nM T79232 CYGN52 42629369 Ki = 28 nM T79232 CEX40M 44215484 Ki = 28 nM T79232 CB82ZC 44232512 IC50 = 490 nM T79232 CBV47F 44243143 Ki = 525 nM T79232 CDI2Q4 44247566 IC50 > 50118.72 nM T79232 CVI6Q3 44275104 Ki = 0.08 nM T79232 CW7JM3 44275447 Ki = 0.8 nM T79232 C08RBM 44279590 Ki = 3981.07 nM T79232 CO92JY 44279908 Ki = 1584.89 nM T79232 CH70NB 44279910 Ki = 1584.89 nM T79232 C2J8GK 44316235 Ki = 24.8 nM T79232 CIE6Y1 44316236 Ki = 276 nM T79232 C24NQS 44316241 Ki = 44.1 nM T79232 CS2ZN9 44321415 Ki = 38.3 nM T79232 CHW9O4 44325345 Ki = 100 nM T79232 CS4UM7 44325362 Ki = 700 nM T79232 C4STM0 44325363 Ki = 1300 nM T79232 C1H6JQ 44325505 Ki = 6400 nM T79232 CAG0C8 44325538 Ki = 4200 nM T79232 CH1P8N 44325558 Ki = 11000 nM T79232 CP4FH8 44325579 Ki = 110 nM T79232 C6OV2D 44325607 Ki = 1900 nM T79232 CZ0BD9 44325689 Ki = 490 nM T79232 C91EAF 44325691 Ki = 250 nM T79232 CO3ZL8 44325695 Ki = 3400 nM T79232 CQ6MC5 44325703 Ki = 30 nM T79232 C1BA7W 44325704 Ki = 1900 nM T79232 C19AEH 44325766 Ki = 410 nM T79232 CD86NE 44325804 Ki = 18 nM T79232 CG8P5Z 44325895 Ki = 290 nM T79232 CM94YJ 44325896 Ki = 1400 nM T79232 CV54FN 44325905 Ki = 14000 nM T79232 C08ETV 44325915 Ki = 14000 nM T79232 C95HKU 44332168 IC50 = 20 nM T79232 CSF89I 44332181 IC50 = 10 nM T79232 C6NW1Z 44332207 IC50 = 16 nM T79232 CF3QT6 44332208 IC50 = 46 nM T79232 CPF97V 44332209 IC50 = 12 nM T79232 CRL53G 44332212 IC50 > 1000 nM T79232 C5N1TG 44332226 IC50 = 15 nM T79232 C4UD2C 44332237 IC50 = 74 nM T79232 CB2VP5 44332238 IC50 = 140 nM T79232 C98OKM 44332239 IC50 = 30 nM T79232 CLJN56 44332261 IC50 > 1000 nM T79232 CA1OL4 44332269 IC50 = 41 nM T79232 C8L7KE 44332272 IC50 = 50 nM T79232 C0S9TC 44332273 IC50 = 10 nM T79232 CGT2A0 44335241 IC50 = 59 nM T79232 C6HO3T 44335329 Ki = 23 nM T79232 CO0EQ9 44335343 IC50 = 35 nM T79232 CZ75ET 44335345 IC50 = 5 nM T79232 C23MCR 44335356 IC50 = 250 nM T79232 C8VWX6 44335386 IC50 = 68 nM T79232 C92YST 44336379 IC50 = 4 nM T79232 C7X3QZ 44336402 IC50 = 7 nM T79232 CDTJ17 44336403 IC50 = 8 nM T79232 CENA29 44336404 IC50 = 65 nM T79232 CM61WN 44336418 IC50 = 7 nM T79232 C7ML9D 44336636 IC50 = 5 nM T79232 CZYV25 44336768 IC50 = 78 nM T79232 CD62CM 44336784 IC50 = 5 nM T79232 C7AU5H 44336791 IC50 = 4 nM T79232 C2IJS5 44336799 IC50 = 4 nM T79232 CJR5B7 44352302 IC50 = 1200 nM T79232 CZ60LX 44352757 IC50 = 440 nM T79232 CM4ZJ0 44352767 IC50 = 160 nM T79232 C9UBG4 44352768 IC50 = 314 nM T79232 CTNY07 44352777 IC50 = 1150 nM T79232 CT3Z9C 44352783 IC50 = 150 nM T79232 CVK34U 44352796 IC50 = 180 nM T79232 CLA4U8 44352804 IC50 = 2010 nM T79232 CNL9F6 44361387 Ki = 22000 nM T79232 C5VCQ0 44361403 Ki = 38000 nM T79232 C38FBJ 44361406 Ki = 36000 nM T79232 CT0ZY3 44361521 Ki = 62000 nM T79232 CMG0N3 44361522 Ki = 12000 nM T79232 CNVI32 44374781 IC50 = 82 nM T79232 COUJ27 44374802 IC50 = 110 nM T79232 CVR8H4 44374839 IC50 = 1740 nM T79232 C6R5FT 44400326 Ki = 148 nM T79232 CLA89W 44400327 Ki = 1492 nM T79232 C91DIF 44400363 Ki = 462 nM T79232 CJ97EG 44400406 Ki = 20 nM T79232 CQOC02 44400407 Ki = 24 nM T79232 C9BH3V 44404614 IC50 = 2 nM T79232 CL53XN 44428401 IC50 > 20000 nM T79232 CCRJ39 44428404 IC50 > 5000 nM T79232 CB12IU 44428407 IC50 > 20000 nM T79232 CU27SN 44428408 IC50 > 20000 nM T79232 C3QW1N 44428411 IC50 > 20000 nM T79232 C0F1NG 44428412 IC50 = 2 nM T79232 C16KRC 44428413 IC50 > 500 nM T79232 CWC18T 44428416 IC50 = 5 nM T79232 C2P6RA 44428417 IC50 = 100 nM T79232 CI70BM 44428418 IC50 = 400 nM T79232 C71DNI 44428419 IC50 = 10 nM T79232 CHC68S 44428420 IC50 = 39 nM T79232 CA2JD4 44428423 IC50 = 405 nM T79232 CVX0L8 44428424 IC50 = 43 nM T79232 C1IY3K 44428425 IC50 = 78 nM T79232 C1A7JT 44428426 IC50 = 54 nM T79232 C9VZM6 44428427 IC50 = 128 nM T79232 CT47FA 44428428 IC50 = 1000 nM T79232 CIOT25 44428429 IC50 = 40 nM T79232 C8FC5N 44428430 IC50 = 41 nM T79232 C4KCH9 44428431 IC50 = 262 nM T79232 CBRW08 44428432 IC50 = 85 nM T79232 C5W0AR 44428487 Ki = 3.39 nM T79232 CQAN10 44428488 Ki = 13.3 nM T79232 C6CHM7 44428489 Ki = 18.2 nM T79232 CC6PL8 44428490 Ki = 26.4 nM T79232 C9SN5A 44428491 Ki = 61 nM T79232 CKX2R3 44428492 Ki = 1.13 nM T79232 CU0FQ4 44428493 Ki = 3.6 nM T79232 CMQ7D4 44428494 Ki = 5.12 nM T79232 CN34FX 44428495 Ki = 6 nM T79232 C98HBS 44428496 Ki = 30 nM T79232 C1EWC9 44428497 Ki = 30 nM T79232 CG3ML0 44428498 Ki < 60 nM T79232 CF2YR6 44428500 Ki < 60 nM T79232 CN3PI1 44428501 Ki = 6100 nM T79232 CG5YV2 44428503 Ki > 600 nM T79232 CDTW25 44428505 Ki > 600 nM T79232 CWA6E3 44428507 Ki = 3.7 nM T79232 CQI7J0 44428509 Ki = 5.58 nM T79232 CW4YN3 44428510 Ki = 7.9 nM T79232 CN8X9D 44428512 Ki = 27.5 nM T79232 C3DHA0 44428514 Ki > 30 nM T79232 C8GQR5 44428516 Ki = 0.27 nM T79232 C6OYI1 44428518 Ki = 0.46 nM T79232 C86CIA 44428520 Ki = 1.17 nM T79232 CQYA65 44428522 Ki = 1.45 nM T79232 C1E5YG 44428529 Ki = 1.19 nM T79232 C6FD3C 44428531 Ki = 1.95 nM T79232 C1X7LF 44428533 Ki = 9 nM T79232 CWA05Z 44428535 Ki = 9.9 nM T79232 C12IZH 44428537 Ki = 0.2 nM T79232 CEY1R8 44428538 Ki = 0.38 nM T79232 CB1S8Y 44428540 Ki = 0.41 nM T79232 CZDB42 44428541 Ki = 0.51 nM T79232 CGV02C 44428542 Ki = 0.66 nM T79232 CPX96C 44428543 Ki = 0.82 nM T79232 CIK0W6 44428544 Ki = 0.93 nM T79232 CXW7P0 44428545 Ki = 4.45 nM T79232 CM4R1C 44428546 Ki < 30 nM T79232 C62YNZ 44428547 Ki = 13 nM T79232 C0K3ZC 44428548 Ki = 33 nM T79232 C0JR4V 44428549 Ki > 12 nM T79232 CH60YJ 44428551 Ki = 1.27 nM T79232 CTQ64N 44428557 Ki = 6.5 nM T79232 CN27YO 44428569 Ki = 1.13 nM T79232 C9OSK3 44428570 Ki = 8.7 nM T79232 CJC3Z2 44428573 Ki > 6 nM T79232 CX6DR5 44428578 Ki > 30 nM T79232 CRN2Q1 44428579 Ki = 179 nM T79232 CS8M2O 44433363 IC50 = 1000 nM T79232 CLBA10 44433367 IC50 = 1000 nM T79232 CCI04H 44433372 IC50 = 1000 nM T79232 C9BDH6 44433375 IC50 = 1000 nM T79232 CIE97C 44434716 IC50 = 7000 nM T79232 CL06GF 44444759 IC50 = 100 nM T79232 CF2U3N 44444760 IC50 = 780 nM T79232 CR8OX5 44444761 IC50 = 40 nM T79232 C1YR6A 44444762 IC50 = 2 nM T79232 CLE7W0 44466239 IC50 > 50118.72 nM T79232 CKA3S0 44467347 IC50 > 50118.72 nM T79232 C4DL5C 44469677 IC50 > 10000 nM T79232 C2N8FY 44520848 Ki = 170 nM T79232 C91HXT 44520849 Ki = 13 nM T79232 C3HP9Y 44520850 Ki = 39 nM T79232 CZ5E2V 44520851 Ki = 17 nM T79232 CMGE92 44520852 Ki = 43 nM T79232 CVA7R2 44520853 Ki = 15 nM T79232 C1U0RY 44520854 Ki = 43 nM T79232 CHE1Y6 44520855 Ki = 30 nM T79232 CCW48G 44520856 Ki = 47 nM T79232 CK7O1L 44520857 Ki = 38 nM T79232 C6TOE7 44520858 Ki = 48 nM T79232 CQF23X 44520859 Ki = 22 nM T79232 CFD98V 44520860 Ki = 57 nM T79232 CJCB39 44520861 Ki = 43 nM T79232 CTVS34 44520862 Ki = 44 nM T79232 CT5A0C 44520863 Ki = 43 nM T79232 CPR8F2 44520864 Ki = 55 nM T79232 CR7Y8G 44520865 Ki = 72 nM T79232 CUN6S2 44520866 Ki = 72 nM T79232 CY61JM 44520867 Ki = 190 nM T79232 CW9RI7 44520868 Ki = 13 nM T79232 CRIF68 44520869 Ki = 59 nM T79232 C1JN3D 44520870 Ki = 230 nM T79232 C8X5FQ 44520871 Ki = 40 nM T79232 CVE5Y7 44571386 Ki = 2.512 nM T79232 CKE3V1 44571387 Ki = 12.59 nM T79232 C27LNY 44571388 Ki = 50.12 nM T79232 C5P0CU 44571389 Ki = 79.43 nM T79232 CV0L4G 44571429 Ki = 3.981 nM T79232 CLI1M9 44571488 Ki = 158.49 nM T79232 CL9SO6 44571489 Ki = 501.19 nM T79232 C0SIU3 44571490 Ki = 1584.89 nM T79232 CC0A4K 44571491 Ki = 25.12 nM T79232 CXI7K6 44571492 Ki = 7943.28 nM T79232 CU1XN0 44571529 Ki = 3981.07 nM T79232 C4LIE5 44571530 Ki = 10000 nM T79232 CFD78Y 44572045 Ki = 794.33 nM T79232 C68RXE 44572047 Ki = 3981.07 nM T79232 C4ZET5 44572048 Ki = 1995.26 nM T79232 CH0Z1M 44572105 Ki = 3981.07 nM T79232 C6D2RB 44572107 Ki = 3.162 nM T79232 CMG70R 44577936 Ki = 525 nM T79232 CZD7E3 44577937 Ki = 270 nM T79232 C0HXR2 44577938 Ki = 44 nM T79232 COP3Q0 44577939 Ki = 1220 nM T79232 C10ZLO 44577981 Ki = 3230 nM T79232 C2WE1A 44577982 Ki = 202 nM T79232 C1E6GX 44577984 Ki = 2410 nM T79232 C6R0AW 44578010 Ki = 432 nM T79232 CLCK14 44579399 Ki = 549 nM T79232 C6OK3X 44579400 Ki > 10000 nM T79232 C0IHE7 44579401 Ki = 3800 nM T79232 CU31MF 44579402 Ki > 10000 nM T79232 CXOJ34 44579441 Ki = 2900 nM T79232 CMW6Q7 44579442 Ki = 214 nM T79232 CM7HN8 44581240 Ki = 50.12 nM T79232 CG68XT 44581241 Ki = 25.12 nM T79232 CC5AT2 44581242 Ki = 15.85 nM T79232 C4FZQ9 44581266 Ki = 50.12 nM T79232 CSZ70I 45103785 Ki > 1000 nM T79232 CK4XM7 45103786 Ki > 5000 nM T79232 C5OSG6 45483182 Ki > 8000 nM T79232 CZBU35 45483183 Ki = 5564 nM T79232 C8GVN6 45483194 Ki > 10000 nM T79232 C6I9KO 45483202 Ki = 709 nM T79232 CQ3BL0 45483203 Ki = 553 nM T79232 CYQ36K 45483204 Ki = 188 nM T79232 CYX27Z 45483235 Ki = 8866 nM T79232 CEIU28 45483236 Ki = 720 nM T79232 C06EOV 45483237 Ki = 33 nM T79232 CUJ8V3 45483238 Ki = 192 nM T79232 C4TZ6D 45483239 Ki = 395 nM T79232 CT9B5J 45483240 Ki = 4926 nM T79232 C45UJI 45483241 Ki = 2600 nM T79232 C75VPW 45483242 Ki = 4803 nM T79232 C7IED0 45483243 Ki = 486 nM T79232 CE5M9W 45483247 Ki > 10000 nM T79232 CY95GV 45483255 Ki = 4963 nM T79232 CWA23E 45483256 Ki = 1268 nM T79232 C4ANR9 45483282 Ki = 4617 nM T79232 CJM89E 45483300 Ki = 6164 nM T79232 CYA3F4 45483320 Ki = 3654 nM T79232 CPYH25 45483321 Ki = 6888 nM T79232 C6CI2W 45483323 Ki = 8734 nM T79232 C02MEC 45483324 Ki = 947 nM T79232 CH73EJ 45483325 Ki = 1257 nM T79232 C6LX7B 46225023 Ki = 127 nM T79232 C48JOB 46225048 Ki = 175 nM T79232 CX2S6L 46225049 Ki = 1840 nM T79232 C70FCZ 46225050 Ki = 734 nM T79232 CIM9Y4 46225051 Ki = 941 nM T79232 CZ36XD 46225079 Ki = 255 nM T79232 CA6DS1 46225080 Ki = 586 nM T79232 COT65W 46225081 Ki = 1000 nM T79232 C53ZIX 46225082 Ki = 522 nM T79232 CFLW87 46225083 Ki > 10000 nM T79232 C7A8DU 46225116 Ki = 1940 nM T79232 C4E8NX 46225117 Ki = 1340 nM T79232 C3W6VI 46225118 Ki = 1680 nM T79232 CT8LO5 46225153 Ki = 719 nM T79232 C98EDC 46233065 Ki = 633 nM T79232 CKET01 46233066 Ki > 5000 nM T79232 C4K7AV 46830094 Ki = 539000 nM T79232 CH4F6K 46830095 Ki > 10000 nM T79232 CNU72P 46830096 Ki = 472000 nM T79232 CS6JV3 46844643 Ki > 4200 nM T79232 C3XYK5 46881859 Ki > 4200 nM T79232 CZRH74 46881860 Ki > 4200 nM T79232 CKR89V 46881861 Ki = 1300 nM T79232 CF56RZ 46881862 Ki = 779 nM T79232 CXV24Z 46881892 Ki > 4200 nM T79232 CI3WD5 46881932 Ki > 4200 nM T79232 C0EMW2 46884414 Ki = 1100 nM T79232 C3FUB6 46884437 Ki = 2300 nM T79232 CM0RI1 46884438 Ki > 10000 nM T79232 C4DP6I 46884439 Ki = 3300 nM T79232 CB3X0J 46884440 Ki = 2000 nM T79232 CXTE54 46884441 Ki > 10000 nM T79232 C27WFG 46884478 Ki = 7200 nM T79232 C3U2WD 46884479 Ki = 12000 nM T79232 CB8WK2 46884480 Ki = 5900 nM T79232 CIS28Y 46890052 Ki = 5.4 nM T79232 CWH0O5 46890053 Ki = 17 nM T79232 CG35DC 46890054 Ki = 105 nM T79232 CQPV07 46890055 Ki = 1.07 nM T79232 CMBS14 46890099 Ki = 5.79 nM T79232 CLFP63 46890100 Ki = 23.5 nM T79232 CRP96J 46890101 Ki = 0.71 nM T79232 CNJB38 46890102 Ki = 51.5 nM T79232 CE84XQ 46890151 Ki = 92.2 nM T79232 C8Y6ET 46890152 Ki = 40.6 nM T79232 C8CXM4 46890153 Ki = 315 nM T79232 CZWV30 46890154 Ki = 52 nM T79232 CY3P8V 46890184 Ki = 86.6 nM T79232 C60CEY 46890185 Ki = 111 nM T79232 CO4CU1 46890186 Ki = 94.6 nM T79232 CJD1S7 46890187 Ki = 443 nM T79232 CLON70 46890214 Ki = 95.4 nM T79232 CN76SA 46890215 Ki = 150 nM T79232 C0AZT4 46890216 Ki = 187 nM T79232 CJ0AM6 46890217 Ki = 5000 nM T79232 C1DG3H 46890258 Ki = 116 nM T79232 CJ2L6D 46890259 Ki = 178 nM T79232 CM70JW 46890260 Ki = 94.4 nM T79232 CQWM92 46890261 Ki = 33.8 nM T79232 CC85GR 46890262 Ki = 62.5 nM T79232 CIC2E8 46890288 Ki = 38.6 nM T79232 CC75DR 46890289 Ki = 49.7 nM T79232 CW38OV 46890290 Ki = 7.1 nM T79232 CHFR58 46890438 Ki = 0.05 nM T79232 CVD95O 46890439 Ki = 65 nM T79232 COE5S9 46890440 Ki = 0.31 nM T79232 C0N1MO 46890484 Ki = 11 nM T79232 CR84PB 46890485 Ki = 0.06 nM T79232 CA7BO2 46890486 Ki = 36 nM T79232 CAR94C 46890487 Ki = 20 nM T79232 C8NGZ1 46890488 Ki = 46 nM T79232 CEM4L1 46890528 Ki = 0.54 nM T79232 C2PYH3 46890529 Ki = 25 nM T79232 CCI0R6 46890530 Ki = 0.6 nM T79232 CF83TS 46890531 Ki = 22.4 nM T79232 C0T5MG 46890569 Ki = 2.6 nM T79232 C1JSF8 46890570 Ki = 2.75 nM T79232 C9QJ5V 46890571 Ki = 3.97 nM T79232 C83LYU 46890572 Ki = 1.03 nM T79232 C1VNK6 46890612 Ki = 0.37 nM T79232 C2XDO1 46890613 Ki = 13.3 nM T79232 CC9E4R 46890614 Ki = 4.42 nM T79232 CCM29N 46890615 Ki = 2.26 nM T79232 C39HAX 46890654 Ki = 0.8 nM T79232 CQUA46 46890655 Ki = 58.9 nM T79232 CLJ2O5 46890656 Ki = 3.8 nM T79232 CEH20W 46890657 Ki = 5000 nM T79232 CC7Y0V 46890706 Ki = 3.78 nM T79232 CIP1L7 46890707 Ki = 0.79 nM T79232 CKQ1Y0 46890708 Ki = 38.9 nM T79232 C02IDZ 46890709 Ki = 0.1 nM T79232 CI9J7N 47177173 Ki = 48 nM T79232 CO9JL6 47177176 Ki = 504 nM T79232 CO4WH0 50941635 Ki = 2511.89 nM T79232 CMPE57 52941704 Ki = 1129 nM T79232 C6U3YN 52947354 Ki = 330 nM T79232 CHX2F3 52947410 Ki = 60 nM T79232 CBDS48 52949017 Ki = 314 nM T79232 C0KBC6 53316694 Ki = 1000 nM T79232 CQ43EC 53316695 Ki = 7943.28 nM T79232 CH47QY 53317994 Ki = 1995.26 nM T79232 CS0Q9A 53323297 Ki = 1995.26 nM T79232 CLK0X6 53323298 Ki = 3162.28 nM T79232 CVB45I 53324622 Ki = 39810.72 nM T79232 C24KRL 53325929 Ki = 6309.57 nM T79232 C01HUJ 53349364 Ki = 70 nM T79232 CK2Y5W 53349471 Ki = 4.4 nM T79232 C4TEY2 53358902 Ki > 10000 nM T79232 C63IVJ 53362154 EC50 = 20.89 nM T79232 C21HMW 53362155 EC50 = 1.1 nM T79232 CF60LM 53362156 EC50 = 69 nM T79232 CGMY47 53362202 EC50 = 11.75 nM T79232 C9V8RI 53362203 EC50 = 1.4 nM T79232 CAL1Y3 53362204 EC50 = 3.548 nM T79232 C6N5EX 53362257 EC50 = 5.7 nM T79232 CS40QD 53362258 EC50 = 1.66 nM T79232 CFWL28 53362259 EC50 = 4.074 nM T79232 CNDR76 53362310 EC50 = 7.943 nM T79232 COUH09 53362311 EC50 = 2.089 nM T79232 C1MU4B 53362312 EC50 = 16 nM T79232 CLRT87 53362368 EC50 = 5.129 nM T79232 CG8J6H 53362369 EC50 = 4.786 nM T79232 CD1N3U 53362370 EC50 = 0.8913 nM T79232 CRY95P 53362428 EC50 = 29.51 nM T79232 C3TFA8 53362429 EC50 = 0.26 nM T79232 C4U1PT 53362430 EC50 = 0.2089 nM T79232 C09KLV 53362488 EC50 = 0.57 nM T79232 CRX54F 53362489 EC50 = 0.8128 nM T79232 C3KCI9 53362490 EC50 = 18 nM T79232 CW32MV 53362546 EC50 = 2.884 nM T79232 C5EG6T 53362547 EC50 = 3.89 nM T79232 CUD9F0 53362548 EC50 = 2.692 nM T79232 CVJ9U2 53362603 EC50 = 1.349 nM T79232 CMY7V4 53362604 EC50 = 2.399 nM T79232 CK9V1G 53362605 EC50 = 0.99 nM T79232 CCRZ83 53362670 EC50 = 1.5 nM T79232 CYK9B3 53362671 EC50 = 2.6 nM T79232 CCK0P6 53362672 EC50 = 10 nM T79232 CYG85M 53362729 EC50 = 0.4898 nM T79232 C1IBT7 53362730 EC50 = 15 nM T79232 CI0F3Y 53362731 EC50 = 14 nM T79232 C3XW1F 53362732 EC50 = 14.45 nM T79232 CYTJ92 53362793 EC50 = 510 nM T79232 CQ9CD8 53362794 EC50 = 29.51 nM T79232 CAN2C1 53362795 EC50 > 1000 nM T79232 CO4UA0 53362796 EC50 = 0.69 nM T79232 C0NSZ5 53362797 EC50 = 11.48 nM T79232 CFJO73 53362798 EC50 = 13.8 nM T79232 C2RSW6 53362849 EC50 = 18.62 nM T79232 C5K9YV 53362850 EC50 = 0.537 nM T79232 CB3AR7 53362851 EC50 = 0.61 nM T79232 C42SJF 53362852 EC50 = 7.244 nM T79232 C8U6LX 53362853 EC50 = 7.4 nM T79232 CH93SM 53362854 EC50 = 7.9 nM T79232 C7RYJ0 53362909 EC50 = 2.2 nM T79232 CKV9D6 53362910 EC50 > 1000 nM T79232 CX9YM6 53362911 EC50 = 10.72 nM T79232 C76TQB 53362913 EC50 = 12 nM T79232 C5XCD8 53362914 EC50 = 7.7 nM T79232 C8N0TX 53362915 EC50 = 10.47 nM T79232 CU9X3P 53362962 EC50 = 12.59 nM T79232 C61CNE 53362963 EC50 = 0.7943 nM T79232 CF30CI 53362964 EC50 = 0.25 nM T79232 C6SB7W 53362965 EC50 = 1.4 nM T79232 C32FZM 53362966 EC50 = 3.2 nM T79232 CJ06TA 53362967 EC50 = 1.585 nM T79232 C6AN7Y 53363015 EC50 = 0.9333 nM T79232 C52IOF 53363016 EC50 = 6 nM T79232 C1SHU3 53363017 EC50 = 38.9 nM T79232 CNA2L1 53364234 Ki = 0.2399 nM T79232 C1S7NG 54580246 Ki = 234.42 nM T79232 COWZ62 54580268 Ki = 15.14 nM T79232 C2Y8TO 54580269 Ki = 5.623 nM T79232 CX07UW 54580270 Ki = 12.59 nM T79232 CT6FL8 54580290 Ki = 288.4 nM T79232 CRM43V 54580291 Ki = 33.88 nM T79232 CXQ31C 54580292 Ki > 10000 nM T79232 CBM07U 54580293 Ki = 7.079 nM T79232 C3L7RP 54580516 Ki = 13 nM T79232 CX1H3Z 54580518 Ki = 231 nM T79232 C1ZOM6 54581243 Ki = 51.29 nM T79232 CL8VJ1 54581265 Ki = 95.5 nM T79232 C7E1YX 54581266 Ki = 109.65 nM T79232 CNB26M 54581267 Ki = 112.2 nM T79232 CXFB64 54581268 Ki = 48.98 nM T79232 C6FNR9 54581298 Ki = 89.13 nM T79232 C2CU4M 54581299 Ki = 2.089 nM T79232 CFO6L7 54581300 Ki = 3.162 nM T79232 C7X4LI 54581307 Ki = 215 nM T79232 CB5R2M 54581528 Ki = 219 nM T79232 CR7GD2 54581529 Ki = 74 nM T79232 CUW8C7 54581530 Ki = 10 nM T79232 CD21EL 54581533 Ki = 289 nM T79232 CE9Z1P 54582268 Ki = 239.88 nM T79232 C4LX9O 54582290 Ki = 56.23 nM T79232 CJZ43P 54582291 Ki = 181.97 nM T79232 CWS8Q3 54582310 Ki = 47.86 nM T79232 C2CQ8N 54582311 Ki = 128.82 nM T79232 C0ZNY9 54582318 Ki = 384 nM T79232 CQ7Z8U 54582526 Ki = 243 nM T79232 C8UN6Y 54582950 IC50 = 2 nM T79232 CRCM14 54583238 Ki = 16.6 nM T79232 C4GNC2 54583264 Ki = 338.84 nM T79232 C9YV3Q 54584201 Ki = 2.951 nM T79232 CHWS35 54584224 Ki = 169.82 nM T79232 CKJ9E2 54584252 Ki = 22.39 nM T79232 CW3Z2F 54584253 Ki = 39.81 nM T79232 C7MP0S 54584254 Ki = 0.2344 nM T79232 C73IGF 54584265 Ki = 69 nM T79232 CX5T1G 54584266 Ki = 246 nM T79232 CIGN05 54584267 Ki = 266 nM T79232 CC49GD 54584268 Ki = 2790 nM T79232 C9N2QH 54584476 Ki = 55 nM T79232 CD1A0H 54584477 Ki = 500 nM T79232 CXPY04 54584478 Ki = 101 nM T79232 CQ9OM0 54585160 Ki = 147.91 nM T79232 C1EIP2 54585191 Ki = 23.99 nM T79232 CQ5J8O 54585219 Ki = 56.23 nM T79232 C5RGO2 54585220 Ki = 26.92 nM T79232 CHR91Z 54585227 Ki = 879 nM T79232 C8YD0H 54585429 Ki = 173 nM T79232 C5N7VS 54585431 Ki = 193 nM T79232 CN3U4G 54586150 Ki = 234.42 nM T79232 C3MLH7 54586172 Ki = 0.5623 nM T79232 CL79ME 54586390 Ki = 49 nM T79232 C1N7LU 54586391 Ki > 1000 nM T79232 C60DIQ 54586392 Ki = 15 nM T79232 C89WPM 54586924 Ki = 30.9 nM T79232 CB90MI 54587127 Ki > 1000 nM T79232 C5T4VS 54587156 Ki = 933.25 nM T79232 C4X8KT 54587187 Ki = 4.898 nM T79232 C7D0MI 54587188 Ki = 17.38 nM T79232 CW04PD 54587189 Ki = 1.66 nM T79232 CJ76VF 56657866 Ki = 30 nM T79232 C3T2HR 56657867 Ki = 13.7 nM T79232 CQG9J6 56657868 Ki = 11.8 nM T79232 C31CRV 56658409 EC50 = 0.15 nM T79232 C6T3VC 56658416 EC50 = 0.23 nM T79232 CF5KG4 56663268 Ki = 0.6166 nM T79232 C6J9OK 56663269 Ki = 4.677 nM T79232 CTC8S3 56663270 Ki = 27.54 nM T79232 C9BA6U 56663271 Ki = 89.13 nM T79232 CGCB51 56663272 Ki = 3.02 nM T79232 CW8NH4 56663273 Ki = 0.2089 nM T79232 CJ5FQ4 56664848 Ki = 57 nM T79232 C5V3ME 56664849 Ki = 107 nM T79232 C3SYC9 56665377 EC50 = 0.14 nM T79232 CM0K3N 56666700 Ki = 18.62 nM T79232 CH4UO0 56666701 Ki = 0.5248 nM T79232 CU8V6N 56666702 Ki = 2.089 nM T79232 CYD7P4 56666703 Ki = 1.778 nM T79232 CQN0G9 56668257 Ki = 217 nM T79232 CU7D3F 56670126 Ki = 7.079 nM T79232 CTA4B5 56670127 Ki = 28.18 nM T79232 C03ETR 56670128 Ki = 0.3715 nM T79232 CL07IK 56671720 Ki = 12.2 nM T79232 CU9DK4 56671721 Ki = 656 nM T79232 CSL0C7 56671723 Ki = 17.3 nM T79232 C2RHD8 56672567 IC50 = 2310 nM T79232 CD9FQ8 56672568 IC50 = 580 nM T79232 CSFT32 56672569 IC50 = 1450 nM T79232 CK9L4C 56672570 IC50 = 3.2 nM T79232 C5KN9R 56673645 Ki = 10.96 nM T79232 C87CMS 56673646 Ki = 169.82 nM T79232 CNO51C 56675150 Ki = 7.6 nM T79232 C8GLI4 56675151 Ki = 25.5 nM T79232 C81PEN 56676958 Ki = 0.03981 nM T79232 C6PDL7 56676959 Ki = 63.1 nM T79232 CS85WE 56676960 Ki = 0.6761 nM T79232 C05JPT 56678446 Ki = 3.9 nM T79232 CN4XD2 56679250 IC50 = 609 nM T79232 C2JSF5 56680282 Ki = 0.5495 nM T79232 C6SEY7 56680283 Ki = 0.182 nM T79232 C83FEJ 56680284 Ki = 0.0955 nM T79232 CN15GL 56680285 Ki = 0.03715 nM T79232 CNZU65 56682530 Ki = 16.8 nM T79232 C9IMV6 56682562 IC50 = 3 nM T79232 CG03CS 56683606 Ki = 0.2512 nM T79232 CH3EM0 56683607 Ki = 1.122 nM T79232 CZE63F 56683608 Ki = 7.079 nM T79232 CAG71L 57391220 Ki = 0.61 nM T79232 C26OTQ 57394727 Ki = 0.63 nM T79232 CFM91W 57399933 Ki = 1.1 nM T79232 CHG37B 57519947 Ki = 530 nM T79232 C0DB5C 57519948 Ki = 8700 nM T79232 C15NPY 57520031 Ki = 4800 nM T79232 C7LF9E 57978135 Ki = 1.4 nM T79232 CXPB73 59429617 Ki = 23 nM T79232 CFN06H 59429650 Ki = 295 nM T79232 C65DNK 59657523 Ki = 0.5 nM T79232 CM7D0N 59657559 Ki = 2 nM T79232 C8DY4C 59657596 Ki = 1 nM T79232 C5FA4G 59657599 Ki = 5 nM T79232 CRSJ24 59657616 Ki = 1 nM T79232 C7TFN1 59657691 Ki = 27 nM T79232 CBTU57 67839485 Ki = 2.28 nM T79232 CD1IQ4 70685417 Ki = 790 nM T79232 CCTZ13 70685423 Ki > 1000 nM T79232 CUD97X 71451749 Ki > 10000 nM T79232 C7BCA6 71451750 Ki > 10000 nM T79232 CJGO63 71451752 Ki > 10000 nM T79232 C8KO3M 71453576 Ki > 10000 nM T79232 CG03VC 71455302 Ki = 1753 nM T79232 C0IZ5N 71457081 Ki = 621 nM T79232 C1Q6RX 71462479 Ki > 10000 nM T79232 CWH6T3 72548703 IC50 = 1.1 nM T79232 C2Y4UX 73348432 Ki = 2.9 nM T79232 C7GDP3 73350017 Ki = 22.5 nM T79232 C8GQK9 73350823 Ki = 5600 nM T79232 CQ8UO2 73351518 Ki = 19.7 nM T79232 CY4IW8 73351519 Ki = 28.1 nM T79232 CG8AD1 73354500 Ki = 63.3 nM T79232 CLMY01 76073634 EC50 > 10 nM T79232 C53VYU 76685194 EC50 = 0.1585 nM T79232 CLF3W5 90285421 EC50 = 0.1259 nM T79232 CL45OR 90672737 EC50 > 100 nM T79232 CI2H0D 90679377 EC50 = 6.5 nM T79232 C8U3HO 90680084 EC50 > 100 nM T79232 C45XGB 90680085 EC50 > 100 nM T79232 CS7DP0 118476369 EC50 = 650 nM T79232 C50MTE 118705579 Ki = 258 nM T79232 C9HX7Z 118705580 Ki = 55300 nM T79232 CR3TZ0 118719818 EC50 > 10000 nM T79232 CFG2V7 118719819 EC50 > 10000 nM T79232 C4J6ZO 118719820 EC50 > 10000 nM T79232 C9B2WS 118719821 EC50 = 85 nM T79232 CAFX95 118719822 IC50 = 1300 nM T79232 CH74ZW 118719823 IC50 = 670 nM T79232 C7QI5K 118719824 IC50 = 17 nM T79232 CAP85S 118719825 IC50 = 55 nM T79232 CDR70N 118719826 IC50 = 1400 nM T79232 CH0WU8 118719827 EC50 = 19 nM T79232 C1OMZ4 118719828 EC50 > 10000 nM T79232 C72LOG 118719829 EC50 = 12 nM T79232 CD0P3Q 118719830 IC50 = 2000 nM T79232 CAKC58 118719831 IC50 = 1800 nM T79232 CIK48G 118719832 IC50 = 3400 nM T79232 CDSK02 118719833 EC50 > 10000 nM T79232 C9GSF2 118719834 IC50 = 1900 nM T79232 CS89AW 118719835 EC50 > 10000 nM T79232 CTWG46 118719836 IC50 = 1400 nM T79232 COQ71F 118719837 IC50 = 880 nM T79232 CT3LR1 118719838 IC50 = 970 nM T79232 CX3R0J 118719839 IC50 = 2200 nM T79232 CT3O7P 118719840 IC50 = 1300 nM T79232 CW2F8P 118719841 IC50 = 3200 nM T79232 CC9ZH4 118719842 IC50 = 270 nM T79232 C0LIH8 118719843 IC50 = 730 nM T79232 CYWM79 118719844 IC50 = 350 nM T79232 CGJ05D 118719845 EC50 = 75 nM T79232 CH3DE8 118720259 IC50 = 390 nM T79232 C3DLZ2 118720260 IC50 = 280 nM T79232 COD37S 118720261 IC50 = 1500 nM T79232 CPNB13 118720262 IC50 = 1300 nM T79232 CW4Q3B 118720263 EC50 > 10000 nM T79232 CI1SA4 118720264 EC50 > 10000 nM T79232 CX2K6O 118720265 IC50 = 990 nM T79232 COHG04 118720266 EC50 > 10000 nM T79232 CL2WY9 118720267 IC50 = 2500 nM T79232 C53KXO 118720268 EC50 > 10 nM T79232 CH2T3S 118720269 IC50 = 1800 nM T79232 C7KCE4 118720270 EC50 > 10000 nM T79232 CEK5A6 118720271 EC50 > 10000 nM T79232 C4OSR7 118720272 EC50 > 10000 nM T79232 C2Z8IG 118720273 IC50 = 300 nM T79232 C3SD1R 118720274 IC50 = 740 nM T79232 CXGF75 118720275 EC50 = 86 nM T79232 CZ96MR 118720276 EC50 > 10000 nM T79232 CM1V0E 118720277 EC50 > 10000 nM T79232 CJB1T7 118720278 IC50 = 1400 nM T79232 C4KHJ3 118720279 EC50 > 10000 nM T79232 C85IJS 118720280 IC50 = 1600 nM T79232 CMK0A4 118720281 EC50 > 10000 nM T79232 C1KPF5 118720282 EC50 = 71 nM T79232 C9XE0M 118720283 IC50 = 480 nM T79232 CXV09J 118720284 IC50 > 10000 nM T79232 C2VF6Q 118720285 IC50 = 1300 nM T79232 CLE5W1 118720286 IC50 = 640 nM T79232 C8QYZ7 118720287 IC50 = 330 nM T79232 CMC18U 118720288 IC50 = 2100 nM T79232 CF1RM4 118720289 IC50 = 380 nM T79232 CTS3Q9 118720290 IC50 = 1200 nM T79232 C3AOC2 118734334 Ki = 19 nM T79232 CT9D1K 118734335 Ki = 48 nM T79232 CBR9L6 118734336 Ki = 550 nM T79232 C2I5VS 118734338 Ki = 870 nM T79232 CKGX38 118734339 Ki = 660 nM T79232 C2T4QR 118734423 Ki = 2830 nM T79232 C3V4SH 118734424 Ki = 6620 nM T79232 C34CEN 118734426 Ki = 3900 nM T79232 CF7MJ6 118734427 Ki = 4990 nM T79232 C0XQ4A 118734428 Ki = 24 nM T79232 CQ9J7L 118734429 Ki = 4 nM T79232 C1G0AS 126705667 EC50 > 100 nM T79232 CZ61LK 127034966 EC50 > 5011.87 nM T79232 CA0SN5 127034967 EC50 > 5011.87 nM T79232 CW7EB6 132559160 Ki = 7040 nM T79232 C3NMS8 132822145 Ki = 6.26 nM T79232 CGI81M 132822146 Ki = 6.75 nM T79232 C1GY2T 135156251 EC50 > 10000 nM T79232 CSP87M 135192889 IC50 = 10970 nM T79232 CA6T5H 135192895 IC50 = 1979 nM T79232 CC09BD 135192928 IC50 = 3811 nM T79232 CWQ30S 135192932 IC50 = 1757 nM T79232 CM0P9E 135192948 IC50 = 4697 nM T79232 CSQ0Y2 135192979 IC50 = 7520 nM T79232 CQI48P 135192983 IC50 = 2885 nM T79232 CS8A2H 135192997 IC50 = 819 nM T79232 CG3JX8 135193003 IC50 = 769 nM T79232 C7GE0F 135399794 Ki > 10000 nM T79232 CHEF49 135399804 Ki > 10000 nM T79232 C1FIH5 135399808 Ki > 10000 nM T79232 CRL41Y 135399831 Ki = 730 nM T79232 C86LKI 135413563 IC50 = 8 nM T79232 CK1U7X 135414270 Ki > 10000 nM T79232 C8SI4F 135414288 Ki = 4940 nM T79232 C9U6OV 135414531 Ki = 511 nM T79232 CVZ9N1 135438362 Ki = 611 nM T79232 CO2J1I 135438380 Ki = 2120 nM T79232 CMH7K6 135438560 Ki = 650 nM T79232 CXV2S0 135438576 Ki > 10000 nM T79232 CD6S8V 135446051 Ki = 510 nM T79232 CS2Z9O 135446053 Ki = 437 nM T79232 CT4GW5 135446078 Ki > 10000 nM T79232 CJ2HL6 135461089 Ki > 10000 nM T79232 CYU6R4 135461099 Ki = 3730 nM T79232 CCI0M9 135461396 Ki = 1103 nM T79232 CFT51M 135466581 Ki = 471 nM T79232 CSNQ01 135468119 Ki > 10000 nM T79232 CFS26I 135469685 Ki = 1180 nM T79232 CYHQ58 135469700 Ki = 176 nM T79232 CK8T6Y 135475778 Ki = 3980 nM T79232 C0DM8J 135475964 Ki = 3215 nM T79232 C3Y5GJ 135475983 Ki > 10000 nM T79232 C4SEV8 135476004 Ki = 133 nM T79232 C3U7PI 135489430 Ki = 1286 nM T79232 CTCL26 135491793 Ki > 10000 nM T79232 CZK63J 135491819 Ki = 94 nM T79232 C9ET1M 135493119 Ki = 65 nM T79232 CD53VT 135502557 Ki > 10000 nM T79232 C3W5GY 135505684 Ki > 10000 nM T79232 C59FZN 135505826 Ki > 10000 nM T79232 C0CPM9 135505845 Ki > 10000 nM T79232 CM26GP 135506374 IC50 = 7 nM T79232 C8QL5H 135508167 Ki = 582 nM T79232 CK6S9M 135510027 Ki > 10000 nM T79232 CLK7Y3 135513039 Ki = 6880 nM T79232 C7P0MW 135520200 Ki > 10000 nM T79232 C8J9EC 135520202 Ki = 596 nM T79232 C4YS7O 135520373 Ki = 3610 nM T79232 C5CDZ0 135520376 Ki = 1390 nM T79232 CG46WC 135520378 Ki > 10000 nM T79232 CB7S3Y 135530014 Ki = 615 nM T79232 CU0WL3 135530164 Ki = 618 nM T79232 CRY3M0 135613341 Ki > 10000 nM T79232 CY12JN 135644174 Ki = 600 nM T79232 CT0A1P 135916059 Ki = 37 nM T79232 CHJ03T 135916060 Ki = 167 nM T79232 CO6G5W 135916061 Ki = 170 nM T79232 C5T1NJ 135916062 Ki > 5000 nM T79232 CAN9M3 135916069 Ki = 18 nM T79232 CH2L4N 135916070 Ki = 27 nM T79232 C32QZC 135997467 Ki > 10000 nM T79232 CO03UG 136961690 Ki = 18 nM T79232 CYA2L4 137189941 Ki = 248 nM T79232 CY64JO 137212769 Ki = 409 nM T79232 CY3E7O 137212770 Ki = 266 nM T79232 C1YN5T 137212771 Ki = 194.7 nM T79232 CI0HQ6 137212772 Ki = 62 nM T79232 C0U2ZG 137212773 Ki = 466 nM T79232 C81USM 137212774 Ki = 449 nM T79232 CHZM41 137212775 Ki = 130 nM T79232 CD2SQ5 137212776 Ki = 64 nM T79232 CNZR50 137631348 EC50 > 100 nM T79232 CSKL70 137632034 EC50 = 0.55 nM T79232 CON47G 137632998 EC50 > 100 nM T79232 CWJO17 137633699 EC50 > 100 nM T79232 CTNY20 137634089 EC50 > 100 nM T79232 CGZ12O 137634607 EC50 = 0.65 nM T79232 C0JLD1 137635522 EC50 = 9 nM T79232 CTK80A 137635922 EC50 > 100 nM T79232 C73GYS 137636048 EC50 > 100 nM T79232 CO2Q1A 137637782 EC50 > 100 nM T79232 C8R7MZ 137637867 Ki = 2.84 nM T79232 CU6F1L 137638040 EC50 > 100 nM T79232 CW2FA1 137639236 EC50 = 0.43 nM T79232 CGHQ73 137639317 EC50 > 100 nM T79232 CKSY39 137639340 EC50 > 100 nM T79232 CS1D6A 137639396 EC50 = 8.2 nM T79232 CD5C8H 137640536 EC50 > 100 nM T79232 CH8DK2 137640630 EC50 > 100 nM T79232 CEWQ40 137641012 EC50 > 100 nM T79232 C8TNJ3 137641033 EC50 > 100 nM T79232 CW8AC7 137642420 Ki = 4.68 nM T79232 CNKR47 137643372 EC50 > 100 nM T79232 C1NYP7 137645401 EC50 = 1.3 nM T79232 CD3NB0 137646127 EC50 > 100 nM T79232 C0IVK7 137647081 EC50 > 100 nM T79232 CNZ60A 137647351 EC50 > 100 nM T79232 CO6DZ8 137647481 EC50 > 100 nM T79232 CFG78N 137648249 EC50 > 100 nM T79232 CM5SI7 137648427 EC50 = 3.9 nM T79232 C92UGK 137648677 EC50 = 2.4 nM T79232 C8F4QJ 137648906 Ki = 78 nM T79232 C61EOM 137649234 EC50 > 100 nM T79232 CMS7U4 137650792 EC50 = 0.5 nM T79232 C34LGF 137651105 EC50 > 100 nM T79232 C94TRJ 137651797 EC50 > 100 nM T79232 CBC95F 137652261 EC50 > 100 nM T79232 CI0QE4 137652597 EC50 = 0.034 nM T79232 CO2S9U 137652605 Ki = 2.06 nM T79232 C41YXQ 137652984 EC50 > 100 nM T79232 C0AT6R 137653368 EC50 > 100 nM T79232 C2TW5S 137653639 EC50 = 0.17 nM T79232 CIF85C 137653770 EC50 > 100 nM T79232 CL9YJ6 137653847 EC50 = 4 nM T79232 CW8G3A 137654006 EC50 > 100 nM T79232 CK73UR 137654009 EC50 = 23 nM T79232 CG1DK7 137654217 EC50 > 100 nM T79232 C2N3TK 137654636 EC50 > 100 nM T79232 CVS36J 137654665 EC50 > 100 nM T79232 C3PSE5 137654909 EC50 > 100 nM T79232 CWN2I1 137654919 EC50 > 100 nM T79232 CB20TQ 137656338 EC50 > 100 nM T79232 CAZL21 137656718 EC50 > 100 nM T79232 C3NM6I 137657345 EC50 = 7.3 nM T79232 CB6FS3 137658004 EC50 > 100 nM T79232 C0C7MG 137658241 EC50 > 100 nM T79232 CWI56Q 137658998 EC50 > 100 nM T79232 CKR3T2 137659747 EC50 > 100 nM T79232 C56UYT 137659822 EC50 = 69 nM T79232 CH19JW 137660341 EC50 = 1.4 nM T79232 C9EDO4 137660579 EC50 > 100 nM T79232 C5EU8T 137661047 EC50 = 0.55 nM T79232 C5V6BP 137661245 EC50 = 8.9 nM T79232 CZ7FL0 137662128 EC50 > 100 nM T79232 CT5D3X 142391767 IC50 = 810 nM T79232 CTO5N4 142391805 IC50 = 1867 nM T79232 C7XTV3 145711714 Ki = 1253 nM T79232 CIY9U2 145949926 Ki = 795.1 nM T79232 C5INL8 145950135 Ki = 6807 nM T79232 C9XH8D 145953061 Ki = 1938 nM T79232 CF5I1P 145953063 Ki = 1910 nM T79232 CS4FG6 145955181 Ki = 250.7 nM T79232 C14WVM 145956003 Ki = 1756 nM T79232 C5C8IL 145956239 Ki = 6250 nM T79232 C6F0CS 145959206 Ki = 642.8 nM T79232 C6AVU4 145959208 Ki = 2095 nM T79232 C3Z9BN 145959348 Ki = 1062 nM T79232 CBP35Y 145959434 Ki = 3343 nM T79232 C63UNT 145960494 Ki = 1954 nM T79232 CIG1P6 145961670 IC50 = 14 nM T79232 C53JQB 145962220 Ki = 1681 nM T79232 CRXH51 145963213 IC50 = 35 nM T79232 CB3TK5 145964151 EC50 > 1000 nM T79232 CY0FL4 145964296 Ki = 573 nM T79232 C9U4FR 145964703 EC50 > 1000 nM T79232 CS40EH 145965644 Ki < 10 nM T79232 CYSP85 145965794 IC50 = 110 nM T79232 CAHB80 145966126 Ki < 10 nM T79232 C3R0NB 145966470 EC50 > 1000 nM T79232 CTC9Q6 145966784 EC50 > 1000 nM T79232 CYIE13 145970269 IC50 = 50 nM T79232 C3H7SY 145970757 Ki = 28 nM T79232 CLN68K 145971236 Ki = 874.1 nM T79232 C43AQD 145971417 Ki = 741 nM T79232 CJF16G 145972114 IC50 = 95 nM T79232 CPY61F 145972843 Ki < 10 nM T79232 CK8HA2 145973088 EC50 > 1000 nM T79232 CI9G0B 145974527 IC50 = 9 nM T79232 CFQ05K 145974615 Ki < 10 nM T79232 CNF1J3 145974638 Ki = 164 nM T79232 C7P6YW 145974697 EC50 > 1000 nM T79232 CXD4H3 145974945 EC50 > 1000 nM T79232 CY2MW6 145975112 EC50 > 1000 nM T79232 CVE64Z 145975166 Ki = 67 nM T79232 CQB98S 145975622 EC50 > 1000 nM T79232 C3XM4U 145975847 EC50 > 1000 nM T79232 CJT06P 145976546 Ki < 10 nM T79232 CQ2IG7 145976595 IC50 = 19 nM T79232 CF14DJ 145976648 Ki = 63 nM T79232 C4B3WF 145976821 EC50 > 1000 nM T79232 C15KIT 145977344 EC50 > 1000 nM T79232 CS5CD6 145977918 Ki = 1075 nM T79232 C8K1EH 145977939 EC50 > 1000 nM T79232 CX16OC 145978563 EC50 > 1000 nM T79232 CT1PI4 145978570 Ki = 34 nM T79232 CTYI46 145978612 Ki > 1000 nM T79232 CK83JH 145978698 EC50 > 1000 nM T79232 C7ZPR6 145981307 Ki = 0.2 nM T79232 C63YEI 145981637 Ki = 0.9 nM T79232 C1XP9S 145986380 Ki = 0.4 nM T79232 C28GTI 145990668 Ki = 1280 nM T79232 CE25VD 145993846 Ki = 0.7 nM T79232 CSB84H 155515636 EC50 > 100000 nM T79232 CI4T0F 155518894 EC50 > 100000 nM T79232 CDN37P 155524296 EC50 > 100000 nM T79232 C2RPD0 155527198 EC50 = 4 nM T79232 CA75ZF 155527876 EC50 > 100000 nM T79232 CYOF34 155532160 EC50 > 10 nM T79232 C8OT1G 155533728 EC50 > 100000 nM T79232 C4ZC5Y 155536940 EC50 = 2.2 nM T79232 C2JH0F 155555127 EC50 > 100000 nM T79232 COX4M3 155565903 EC50 > 10 nM T79232 D00HAJ 73347136 IC50 = 740 nM T79232 D00NIT 9810140 Ki = 0.62 nM T79232 D00SGZ 9917025 Ki = 0.3 nM T79232 D01WHI 135413562 Ki = 0.65 nM T79232 D09RIE 44419028 Ki = 151 nM T79232 D0K5NV 44428109 Ki = 2.1 nM T79232 D0L0RP 44428107 Ki = 0.09 nM T79232 D0NC8V 6918854 Ki < 6309.57 nM T79232 D0Q0OR 10461270 Ki = 143 nM T79232 D0Q3VN 44428111 Ki = 0.032 nM T79232 D0R7QC 44419039 Ki = 54.2 nM T79232 D0T4ML 5311202 Ki = 3200 nM T79232 D0W3IQ 44419025 Ki = 11.4 nM T79232 D0ZD0W 11366713 Ki = 88 nM T82083 D01BYB 5957 EC50 = 43000 nM T82083 D07QQP 10219163 EC50 = 800 nM T82083 D0H2UB 5361 EC50 > 100000 nM T82083 D0S6AE 148197 EC50 = 130 nM T82083 D0Z7FU 6133 EC50 = 39 nM T82083 C9K3IP 78253 IC50 > 10000 nM T82083 CS2M9I 148196 EC50 = 130 nM T82083 C6VB7R 150973 EC50 > 100000 nM T82083 CM6QD5 189010 EC50 = 4640 nM T82083 CO6A2E 451388 EC50 = 3900 nM T82083 C9QSK6 3018777 IC50 > 10000 nM T82083 C7NR6U 3081495 EC50 > 100000 nM T82083 C6P7VU 5311303 EC50 > 100000 nM T82083 C5OT9B 6604161 IC50 = 625 nM T82083 CRK8Q6 9853990 EC50 = 80 nM T82083 CVZX40 9875011 EC50 = 870 nM T82083 CR4UQ9 9875516 EC50 = 140 nM T82083 CM96ZK 10168108 EC50 > 20000 nM T82083 CI9K1V 10191162 EC50 = 4233 nM T82083 CO0L9C 10234467 EC50 > 10000 nM T82083 C7OK5W 10255482 EC50 = 600 nM T82083 CM4K6R 10303040 EC50 = 4121 nM T82083 CF08GK 10432343 EC50 = 3500 nM T82083 CMW2L8 10929115 EC50 = 49 nM T82083 COI83E 11525909 EC50 = 1200 nM T82083 C9M1FO 11534074 EC50 >= 100000 nM T82083 CZ8C1X 11606036 EC50 > 100000 nM T82083 C2XOC1 11993883 EC50 > 100000 nM T82083 COZ6Y2 11993885 EC50 > 100000 nM T82083 CH4XG1 11993887 EC50 > 100000 nM T82083 CZ1J9L 11993889 EC50 > 100000 nM T82083 CQ9ZE4 11993891 EC50 = 3990 nM T82083 C3NZ6K 11994005 EC50 > 100000 nM T82083 CNBZ84 11994007 EC50 > 1000 nM T82083 CN0HI1 11994009 EC50 > 100000 nM T82083 CI48FW 11994013 EC50 > 100000 nM T82083 C2MD3V 11995641 EC50 > 100000 nM T82083 CM59TJ 11995643 EC50 > 100000 nM T82083 C2B6HY 16082731 EC50 = 3100 nM T82083 CR6W9O 16216480 EC50 > 20000 nM T82083 C3ZEI4 16655024 EC50 > 100000 nM T82083 C1QCG8 23379800 EC50 = 7200 nM T82083 C7GV8K 23662455 IC50 = 1700 nM T82083 CYZK58 23664788 IC50 = 2760 nM T82083 C8KY2H 23668635 IC50 = 3580 nM T82083 CN5OC4 23673110 IC50 = 3160 nM T82083 CA08ML 23674540 IC50 = 3490 nM T82083 CK5S9W 23686655 IC50 = 2820 nM T82083 C4HJO0 23718715 IC50 = 7180 nM T82083 C20IDU 24857827 EC50 = 710 nM T82083 CHA2I6 24868313 IC50 = 7420 nM T82083 CNLM45 44152334 IC50 = 11200 nM T82083 C5WP3I 44157464 IC50 = 1450 nM T82083 CTZ81X 44157465 IC50 = 1180 nM T82083 CJN39O 44157467 IC50 = 14400 nM T82083 CJ4E6Y 44157518 IC50 = 3450 nM T82083 C3CU9F 44415751 EC50 > 100000 nM T82083 C9HSG4 44417696 EC50 = 2920 nM T82083 C69SHE 44417704 EC50 > 100000 nM T82083 C28AEV 44420650 EC50 = 8300 nM T82083 C2D1MQ 44439743 EC50 = 7043 nM T82083 CW2U7Z 44439757 EC50 = 3583 nM T82083 C42YBU 44439758 EC50 = 20000 nM T82083 C0IBA3 44439765 EC50 > 20000 nM T82083 CEYV61 44456046 IC50 = 1910 nM T82083 C1DU4Z 44456078 IC50 = 2340 nM T82083 CHF3N0 44456160 IC50 = 3530 nM T82083 CLN38C 44456165 IC50 = 2630 nM T82083 C1W8IK 44456201 IC50 = 2220 nM T82083 CD50FC 44457390 EC50 > 100000 nM T82083 C6Z7JE 44457427 EC50 = 400 nM T82083 C41BAQ 44583493 IC50 = 6100 nM T82083 CD5O7G 44583580 IC50 = 10000 nM T82083 C9BM5G 44583581 IC50 > 10000 nM T82083 C84HQM 44585515 EC50 > 10000 nM T82083 C8Q2EX 44585516 EC50 = 4780 nM T82083 C0S8XM 44585517 EC50 = 6300 nM T82083 C1V5YQ 44585518 EC50 = 2060 nM T82083 C9JU8Z 44585519 EC50 = 1770 nM T82083 C09XZT 44585520 EC50 > 10000 nM T82083 CRS2E1 44585521 EC50 = 4320 nM T82083 CD9A6E 44585986 EC50 = 8110 nM T82083 CR0W7K 44585987 EC50 = 90 nM T82083 CUPC35 44585988 EC50 = 5350 nM T82083 CW93JX 44586005 EC50 = 4640 nM T82083 C3RS8O 44586006 EC50 = 7930 nM T82083 CALX92 44586007 EC50 = 1260 nM T82083 CJHP17 44586025 EC50 = 5520 nM T82083 COB6E3 44586026 EC50 = 280 nM T82083 CR57TZ 44586027 EC50 = 5270 nM T82083 CV1MB6 44586042 EC50 = 2700 nM T82083 C5JV6T 44586043 EC50 = 2530 nM T82083 C08CEM 44586044 EC50 = 1960 nM T82083 C3R4LJ 44586045 EC50 = 1120 nM T82083 CIA68B 44602426 EC50 > 100000 nM T82083 CNDO30 45104519 EC50 >= 20000 nM T82083 CG7VB4 45141594 IC50 > 100000 nM T82083 CC06FN 45141778 IC50 > 100000 nM T82083 C12QZE 45485253 EC50 = 6450 nM T82083 CKJ8L5 46228661 IC50 = 1940 nM T82083 CH6F5O 46228691 IC50 = 4040 nM T82083 CI4QC0 46228692 IC50 = 3300 nM T82083 CHI0N8 46228790 IC50 = 30000 nM T82083 CX01WL 46228816 IC50 > 100000 nM T82083 CS8I2W 46830491 EC50 = 790 nM T82083 C25PCZ 46830492 EC50 = 560 nM T82083 C2Q0RG 46831384 EC50 = 180 nM T82083 CN26KT 46831386 EC50 = 6230 nM T82083 C0B9RN 46831686 EC50 = 1150 nM T82083 CS1D6Q 46831692 EC50 = 25 nM T82083 CJQ84K 46890063 EC50 = 300 nM T82083 C0X7QY 46890111 EC50 = 85 nM T82083 C7QD6O 51050128 IC50 = 1510 nM T82083 C0OL1Z 51050130 IC50 = 9250 nM T82083 CEGF57 51050132 IC50 = 1390 nM T82083 C9DN0M 51050133 IC50 = 30000 nM T82083 CNYH17 51050134 IC50 = 12500 nM T82083 CPCQ79 51050233 IC50 > 10000 nM T82083 CW0N3F 52952183 EC50 > 100000 nM T82083 CK8YW6 52952280 EC50 = 1520 nM T82083 CWR0B6 52952281 EC50 = 4900 nM T82083 CHC4O2 52952282 EC50 = 5980 nM T82083 CZ86FL 52952283 EC50 >= 100000 nM T82083 C2DZ5A 52952391 EC50 = 4490 nM T82083 CA8JY6 52952392 EC50 >= 100000 nM T82083 C2GNH6 52952393 EC50 >= 100000 nM T82083 C2IA6G 52952394 EC50 > 100000 nM T82083 C0MWH4 52952395 EC50 = 4330 nM T82083 CZO8K6 52952396 EC50 > 100000 nM T82083 C67NQB 52952397 EC50 > 100000 nM T82083 CBL7S0 52952494 EC50 > 100000 nM T82083 CLGF37 52952495 EC50 > 100000 nM T82083 CA3CS6 52952496 EC50 > 100000 nM T82083 CVO0A1 52952497 EC50 = 7300 nM T82083 C15FQS 52952603 EC50 = 7870 nM T82083 CHR9Q8 52952604 EC50 = 3930 nM T82083 C8FUJ5 53262904 EC50 = 62 nM T82083 CA1L7N 53308118 IC50 = 10000 nM T82083 C2JIO7 53308272 EC50 = 97 nM T82083 CDH9J7 53308826 EC50 = 210 nM T82083 CJZI31 53308961 EC50 = 2110 nM T82083 CG9X8W 53309242 EC50 = 2540 nM T82083 CNLP93 53309244 EC50 = 183 nM T82083 CYQ90K 53309245 EC50 = 4480 nM T82083 CR3DH9 53309379 EC50 = 620 nM T82083 C21ZMJ 53309380 EC50 = 910 nM T82083 CGJ86N 53309381 EC50 = 227 nM T82083 C4HL7B 53309528 EC50 = 670 nM T82083 CDN2V9 53309529 EC50 = 310 nM T82083 CI4G5S 53309530 EC50 = 220 nM T82083 CEK7Y6 53318846 IC50 = 6450 nM T82083 C65QBU 53320148 IC50 = 6960 nM T82083 C98MFN 53326684 IC50 = 10000 nM T82083 CGV02T 54584406 EC50 = 1100 nM T82083 C7ANP0 56944330 IC50 = 3210 nM T82083 C2F3LX 70694098 EC50 = 9400 nM T82083 CTEL13 71459956 EC50 > 30000 nM T82083 CH0O5B 71459957 EC50 > 20000 nM T82083 CF61BN 71459959 EC50 > 30000 nM T82083 C6K4MB 71531031 IC50 = 2200 nM T82083 CAS84P 76324375 EC50 > 100000 nM T82083 C3P1MQ 90656210 EC50 = 470 nM T82083 C6CEH7 90656211 EC50 = 54 nM T82083 CVOB74 90656212 EC50 = 430 nM T82083 CL2VA3 90656213 EC50 = 100 nM T82083 C6R2QF 90656214 EC50 = 105 nM T82083 C6PS8Q 90656215 EC50 = 141 nM T82083 CE32XG 90656216 EC50 = 114 nM T82083 CX53VO 90656217 EC50 = 91 nM T82083 C4W0IB 90656218 EC50 = 95 nM T82083 C1AD7F 90656219 EC50 = 84 nM T82083 CL9XR5 90656220 EC50 = 23 nM T82083 C93EMP 90656221 EC50 = 300 nM T82083 CJ80KG 90656222 EC50 = 250 nM T82083 CPH41T 90656223 EC50 = 20 nM T82083 CBGQ40 90656224 EC50 = 410 nM T82083 CA3X6O 90656225 EC50 = 128 nM T82083 C5VWX0 90656226 EC50 = 47 nM T82083 CFCU65 90656227 EC50 = 40 nM T82083 C5FE0D 90656230 EC50 = 70 nM T82083 C4F9RY 90656231 EC50 = 93 nM T82083 C57TEN 90656232 EC50 = 1330 nM T82083 CS7WF2 90666789 EC50 > 10000 nM T82083 CE0XU1 90666790 EC50 = 352 nM T82083 C32TOB 90666791 EC50 = 7440 nM T82083 CNV09R 90666793 EC50 = 2200 nM T82083 CSE39Z 90666794 EC50 = 952 nM T82083 C40LJI 90666798 EC50 = 636 nM T82083 C4HT6U 90666802 EC50 = 3300 nM T82083 CHIG78 132574706 IC50 = 482 nM T82083 CA5LF2 135528590 EC50 = 540 nM T82083 CEA7D5 136169604 IC50 = 73000 nM T82083 CBF83D 137631394 IC50 = 21100 nM T82083 C6ZB1D 137632198 IC50 = 746 nM T82083 C8DGS4 137633744 IC50 = 1760 nM T82083 CJ9O1V 137635546 IC50 = 2990 nM T82083 CD3LZ2 137635749 IC50 = 4980 nM T82083 CE4V1S 137639206 IC50 > 30000 nM T82083 CV2IZ1 137639602 IC50 = 4130 nM T82083 CP1N8K 137640480 IC50 = 1690 nM T82083 C4GA0J 137641946 IC50 = 409 nM T82083 C7O3US 137643396 IC50 = 233 nM T82083 CD1JE8 137644032 IC50 = 1540 nM T82083 CPT2Q0 137645875 IC50 = 9340 nM T82083 C3ZNA5 137647423 IC50 = 3370 nM T82083 CQ0M7L 137648293 IC50 = 100000 nM T82083 CUR8V1 137648798 IC50 = 395 nM T82083 CJMX73 137648855 IC50 = 1650 nM T82083 CU7G2K 137651974 IC50 > 100000 nM T82083 C2PX1Y 137654054 IC50 > 30000 nM T82083 C1SX8J 137654771 IC50 = 373 nM T82083 CUEQ97 137659976 IC50 > 30000 nM T82083 C6MG8A 90656228 EC50 = 200 nM T82083 D01ZZJ 49867142 EC50 = 4980 nM T82083 D02HAL 6031 EC50 = 14000 nM T82083 D04IWB 10174453 EC50 = 350 nM T82083 D05MXI 42611190 IC50 > 10000 nM T82083 D06DBA 23680506 IC50 = 2590 nM T82083 D06GQY 91934096 IC50 > 10000 nM T82083 D06PIW 53262902 EC50 = 23 nM T82083 D07LYU 53262890 EC50 = 73 nM T82083 D07QYU 4881 EC50 > 10000 nM T82083 D07TSE 16082712 EC50 > 1000 nM T82083 D08DXA 23675622 IC50 = 1970 nM T82083 D0B0ZQ 9875920 IC50 = 1140 nM T82083 D0DZ1K 45141593 IC50 > 10000 nM T82083 D0GF4I 3033941 EC50 = 23 nM T82083 D0P0EP 161647 EC50 > 100000 nM T82083 D0P4GP 52952605 EC50 = 9300 nM T82083 D0P7RI 9872620 EC50 = 3460 nM T82083 D0Q1HE 16116566 EC50 = 2400 nM T82083 D0T4WF 11994011 EC50 > 100000 nM T82083 D0UC4G 25090818 IC50 = 3980 nM T94880 D03ZBT 11626560 IC50 > 100 nM T94880 D0E3TC 44259 IC50 = 2.75 nM T94880 D0O6WV 24794418 IC50 = 4.3 nM T94880 D03BNU 59604787 IC50 > 10000 nM T94880 D03RHV 72793043 IC50 = 4060 nM T94880 D08OEW 72792975 IC50 = 390 nM T94880 D0M9TR 72793042 IC50 = 4910 nM T94880 CACS26 11561968 Ki > 2000 nM T94880 CU0E8O 11690457 Ki > 2000 nM T94880 C5VPH9 16129448 IC50 = 1030 nM T94880 CF57GK 46215462 IC50 = 17 nM T94880 CLS29B 46872626 IC50 > 10000 nM T94880 C3V5XE 53355503 IC50 = 48 nM T94880 CC62KV 54915268 IC50 > 30000 nM T94880 C0MYE4 56947174 IC50 = 670 nM T94880 C1MR8Q 60097495 IC50 > 1000 nM T94880 C9ZCT2 62705065 IC50 > 1000 nM T94880 C10AMI 66553589 IC50 > 10000 nM T94880 C37NKO 67129970 IC50 = 3210 nM T94880 CK80LJ 67130050 IC50 = 4140 nM T94880 CV63UL 67240318 IC50 > 10000 nM T94880 CJLT43 67471113 IC50 = 1400 nM T94880 CXR9Y0 68212353 IC50 = 1500 nM T94880 CEH69L 68212361 IC50 = 410 nM T94880 C4V3DJ 68212395 IC50 = 120 nM T94880 CPZ8D7 68212421 IC50 = 250 nM T94880 CBUE63 68212479 IC50 = 11000 nM T94880 CR0B8N 68212480 IC50 = 14 nM T94880 CZJ83X 68212482 IC50 = 2.9 nM T94880 C1QXE9 68212489 IC50 = 450 nM T94880 C5H8DO 68212494 IC50 = 17000 nM T94880 C2WDO9 68212498 IC50 = 370 nM T94880 C7PT2D 68212505 IC50 = 22 nM T94880 CKPF54 68212509 IC50 = 5.9 nM T94880 C40GFP 68212528 IC50 > 30000 nM T94880 CJY4P6 68212724 IC50 = 260 nM T94880 C2ZCD6 68212733 IC50 = 370 nM T94880 C4ARE2 68212746 IC50 = 75 nM T94880 CTM2R4 68212750 IC50 = 5400 nM T94880 C5MG7K 68212755 IC50 = 80 nM T94880 COV36W 68212757 IC50 = 71 nM T94880 C51DUT 68212759 IC50 = 18 nM T94880 CL95KS 68212760 IC50 = 2800 nM T94880 CQD3H2 68212763 IC50 = 4300 nM T94880 C6GU4S 68212779 IC50 > 30000 nM T94880 CG5VP7 68212780 IC50 = 13000 nM T94880 CJR90K 68212791 IC50 = 340 nM T94880 CS5C0R 68212798 IC50 = 60 nM T94880 C7GRV2 68755406 IC50 > 10000 nM T94880 CO4F8Q 70681237 IC50 = 380 nM T94880 C36TJD 70681238 IC50 = 85 nM T94880 CZVD75 70681239 IC50 = 50 nM T94880 C4DT3L 70681245 IC50 = 10000 nM T94880 C2B8DE 70681768 IC50 > 30000 nM T94880 CQAU72 70681769 IC50 = 2100 nM T94880 CG80HU 70681780 IC50 = 150 nM T94880 CX2W7Y 70683322 IC50 = 380 nM T94880 CCJA41 70683323 IC50 > 50000 nM T94880 CL9RI4 70683324 IC50 = 110 nM T94880 CNAC18 70683325 IC50 = 340 nM T94880 CG3E2S 70683326 IC50 = 50 nM T94880 CM3ZE4 70683327 IC50 = 60 nM T94880 CG28BF 70683336 IC50 = 100 nM T94880 CK5I0P 70685426 IC50 = 1400 nM T94880 CUC73G 70685427 IC50 = 60 nM T94880 CPOI37 70685428 IC50 = 100 nM T94880 C3IKD0 70685429 IC50 = 42 nM T94880 CG94HD 70685430 IC50 = 40 nM T94880 CKU02L 70685438 IC50 = 20 nM T94880 C8JYH4 70686029 IC50 = 75000 nM T94880 C1TY5D 70687566 IC50 = 120 nM T94880 CK4S0N 70687567 IC50 = 490 nM T94880 C9Q1CO 70687568 IC50 = 28 nM T94880 CT15YD 70687569 IC50 = 67 nM T94880 CKG63T 70687570 IC50 = 30 nM T94880 C0GVD6 70687571 IC50 = 50 nM T94880 C92FQP 70687572 IC50 = 60 nM T94880 C6U2WZ 70687578 IC50 = 20 nM T94880 CZ6YA9 70691762 IC50 = 2600 nM T94880 C5J3CU 70691763 IC50 = 34 nM T94880 CN1SQ4 70691764 IC50 = 40 nM T94880 COP3Z0 70691765 IC50 = 40 nM T94880 C7LVS2 70692345 IC50 = 77 nM T94880 CZ6E4M 70693824 IC50 = 2400 nM T94880 CH9E2Q 70693825 IC50 = 340 nM T94880 C56RZU 70693834 IC50 = 60 nM T94880 CWP13X 70695379 IC50 > 30000 nM T94880 C2IH6R 70695946 IC50 = 1900 nM T94880 C3KNG1 70695947 IC50 = 640 nM T94880 CD6M8K 70695948 IC50 = 400 nM T94880 C3H8PZ 70695949 IC50 = 80 nM T94880 CM0D3O 70696465 IC50 > 30000 nM T94880 CTB5O3 70696471 IC50 = 640 nM T94880 C5Q3YE 70697396 IC50 > 30000 nM T94880 CH0B8N 70789756 IC50 = 400 nM T94880 C0E2FS 71552533 IC50 = 4200 nM T94880 CC6N4S 71552534 IC50 = 7200 nM T94880 CBF79Y 71552535 IC50 = 1100 nM T94880 CTK2E9 71552536 IC50 = 810 nM T94880 C4NKR0 71552618 IC50 = 2000 nM T94880 CEBK17 71552619 IC50 = 1100 nM T94880 CO6UE9 71552620 IC50 = 260 nM T94880 CQI0T6 71552621 IC50 = 110 nM T94880 C4PR9X 71552622 IC50 = 180 nM T94880 C97SFB 71552692 IC50 = 170 nM T94880 CBY0V2 71552693 IC50 = 360 nM T94880 C7E2VT 71552694 IC50 = 200 nM T94880 CT6GM8 71552695 IC50 = 37 nM T94880 CA3O6K 71552696 IC50 = 270 nM T94880 CQW4X1 71552779 IC50 = 68 nM T94880 CG9C3F 71552780 IC50 = 35 nM T94880 CR3D6A 71552781 IC50 = 2100 nM T94880 C8RD2U 71552782 IC50 = 9500 nM T94880 CBC7A1 71552783 IC50 = 11200 nM T94880 CW4F5I 71552784 IC50 = 11200 nM T94880 C0PB4E 71552866 IC50 = 850 nM T94880 C2IC5R 71552867 IC50 = 9700 nM T94880 C14MFN 71552868 IC50 = 3000 nM T94880 CGR91F 71552869 IC50 = 1580 nM T94880 CJ48FQ 71552940 IC50 = 215 nM T94880 C1NPL0 71552941 IC50 = 355 nM T94880 CA4PS8 71552942 IC50 = 70 nM T94880 CU2EL6 71553007 IC50 = 160 nM T94880 C0EC4Z 71553008 IC50 = 380 nM T94880 CPME80 71553009 IC50 = 1300 nM T94880 CK6CP5 71553010 IC50 = 500 nM T94880 C3UA9C 71553011 IC50 = 520 nM T94880 CEZ15Y 71553012 IC50 = 270 nM T94880 CF1LY3 71553083 IC50 = 190 nM T94880 C1CM5E 71553084 IC50 = 41 nM T94880 CVIA91 71553085 IC50 = 2 nM T94880 CQ91EB 71553086 IC50 = 9 nM T94880 CZM0S4 71553087 IC50 = 6 nM T94880 CJCE72 71553151 IC50 = 3 nM T94880 C1TR3O 71553152 IC50 = 10 nM T94880 CH08XN 71553153 IC50 = 92 nM T94880 CEN63Z 71553155 IC50 = 44 nM T94880 CQZ8D4 71553156 IC50 = 150 nM T94880 C5YN8K 71553236 IC50 = 15 nM T94880 C1BCX0 71579696 IC50 > 1000 nM T94880 CS1H6O 71717919 IC50 = 1900 nM T94880 C4Q2HC 71721525 IC50 = 250 nM T94880 CQ3JN8 71819732 IC50 = 630 nM T94880 C9NVM8 72192165 IC50 = 280 nM T94880 C7A8XR 72547635 IC50 > 30000 nM T94880 CUPN10 72547636 IC50 = 16200 nM T94880 C5MI7D 72547637 IC50 = 1200 nM T94880 CD93WQ 72547638 IC50 = 1700 nM T94880 C49RTS 72547864 IC50 > 30000 nM T94880 C45UFT 72547868 IC50 = 2300 nM T94880 CM23ZS 72548104 IC50 = 4300 nM T94880 CO7MN3 72548105 IC50 > 30000 nM T94880 CH05EK 72551069 IC50 = 2200 nM T94880 C07THM 72551070 IC50 = 900 nM T94880 CVNK29 72551073 IC50 = 400 nM T94880 CO3UW2 72551074 IC50 = 530 nM T94880 CP09RS 72792559 IC50 > 30000 nM T94880 C3PTC7 72792560 IC50 = 810 nM T94880 C12IMZ 72792561 IC50 = 390 nM T94880 C2E0RN 72792562 IC50 = 36 nM T94880 CZXU21 72792563 IC50 = 21 nM T94880 CD7UM4 72792564 IC50 = 28 nM T94880 C38OCL 72792627 IC50 = 24 nM T94880 C39PHS 72792906 IC50 = 94 nM T94880 C6HYA4 72792907 IC50 = 24 nM T94880 C16ETP 72792908 IC50 = 33 nM T94880 CNSX89 72792909 IC50 = 21 nM T94880 C7HXN3 72792910 IC50 > 30000 nM T94880 CGP01I 72792971 IC50 = 84 nM T94880 CXNF57 72792972 IC50 = 58 nM T94880 CGDL83 72792973 IC50 = 280 nM T94880 CJGF34 72792974 IC50 = 430 nM T94880 C4N9TK 72792977 IC50 = 1340 nM T94880 C5B9CI 72793044 IC50 > 30000 nM T94880 C86UHM 72793045 IC50 > 30000 nM T94880 C75QHA 72793046 IC50 = 6850 nM T94880 C1MPN7 72793047 IC50 = 2580 nM T94880 CRJ81Y 72793048 IC50 = 1590 nM T94880 CL9EA5 72793105 IC50 = 440 nM T94880 CVT7A9 72793106 IC50 = 370 nM T94880 C39VXU 72793107 IC50 > 30000 nM T94880 C43SNK 72793108 IC50 > 30000 nM T94880 C9XAE8 72793109 IC50 = 1160 nM T94880 CZA34R 72793110 IC50 = 300 nM T94880 CU9R4X 72793111 IC50 = 80 nM T94880 CD2K0R 72793177 IC50 = 8940 nM T94880 CP26TN 72793178 IC50 = 6140 nM T94880 CKV95R 72793179 IC50 = 2930 nM T94880 CH80BD 72793182 IC50 > 30000 nM T94880 CAJ65L 72793183 IC50 > 30000 nM T94880 CVR1I4 72793252 IC50 = 6700 nM T94880 CJWB46 72793253 IC50 > 30000 nM T94880 CMIH15 72793254 IC50 > 30000 nM T94880 C30IXP 72793255 IC50 = 190 nM T94880 C6YFO5 72793256 IC50 = 480 nM T94880 CJG79M 72793257 IC50 = 540 nM T94880 CK6U5Z 72793332 IC50 = 370 nM T94880 CI6JX5 72793333 IC50 = 17900 nM T94880 CA4ET8 72793334 IC50 = 660 nM T94880 C6JW5N 72793335 IC50 = 830 nM T94880 CROW51 72793336 IC50 = 1500 nM T94880 C65KJA 72793337 IC50 = 450 nM T94880 C7IA8R 72793397 IC50 = 240 nM T94880 CD85ZE 72793399 IC50 = 700 nM T94880 CI4E7H 72793400 IC50 = 570 nM T94880 C02GET 72793401 IC50 > 30000 nM T94880 C9WYE4 72793466 IC50 = 620 nM T94880 C37FKG 72793468 IC50 = 2000 nM T94880 COU2I8 72793469 IC50 = 19500 nM T94880 C49MHY 72793532 IC50 = 2000 nM T94880 C3K2BV 72793533 IC50 = 4100 nM T94880 C5UH4O 72793534 IC50 > 30000 nM T94880 C2Z6FI 72793535 IC50 > 30000 nM T94880 CLTB82 72793536 IC50 > 30000 nM T94880 CQ7KX1 72793601 IC50 = 170 nM T94880 CW0PY4 72793602 IC50 = 11700 nM T94880 CKB3O6 72793603 IC50 > 30000 nM T94880 CI9L8K 72793604 IC50 > 30000 nM T94880 CMD9F8 72793605 IC50 = 270 nM T94880 CE60AT 72793606 IC50 = 88 nM T94880 C75UBS 72793607 IC50 = 110 nM T94880 C51VIE 72793608 IC50 = 21900 nM T94880 COL6Y5 72793609 IC50 = 940 nM T94880 CJ9C7M 72793610 IC50 = 5100 nM T94880 CGCL01 72793611 IC50 = 6700 nM T94880 CZ5QY9 72793612 IC50 > 30000 nM T94880 CJ87CG 73211763 IC50 = 100 nM T94880 CVNW01 73386831 IC50 > 1000 nM T94880 C1V3NZ 73425588 IC50 = 5.83 nM T94880 CQ4ZH2 74538669 IC50 = 220 nM T94880 CG7VE4 76309971 IC50 = 1600 nM T94880 C17BGH 76328134 IC50 = 1370 nM T94880 CHIZ70 89495685 IC50 = 17 nM T94880 CS6IA4 89495748 IC50 = 45 nM T94880 CW1OS0 89495775 IC50 = 33 nM T94880 CL2DH6 118433464 IC50 = 10 nM T94880 C01OAD 118433470 IC50 = 29 nM T94880 C9ENZ0 118433703 IC50 = 34 nM T94880 CQU1R4 118443520 IC50 = 13 nM T94880 C8OSQ4 118443521 IC50 = 6.7 nM T94880 CAM76F 118443524 IC50 = 6.9 nM T94880 C3DEP2 118443546 IC50 = 12 nM T94880 CGO6B1 118443548 IC50 = 151 nM T94880 CADG96 118443549 IC50 = 12 nM T94880 CM92EG 118443553 IC50 = 6.7 nM T94880 CVWR20 118443556 IC50 = 99 nM T94880 CC9FK0 118443560 IC50 = 4.3 nM T94880 CRZ68N 118443583 IC50 = 4.4 nM T94880 C9I5MC 118443585 IC50 = 26 nM T94880 CE42TF 118443586 IC50 = 850 nM T94880 C5YJT1 118443594 IC50 = 3.4 nM T94880 CL0YO5 118443595 IC50 = 3.1 nM T94880 CG3K5V 118443597 IC50 = 33 nM T94880 C12WAU 118446433 IC50 = 1662 nM T94880 CFBY13 118446434 IC50 = 22 nM T94880 CY6C1E 122179442 IC50 > 10000 nM T94880 CG0RP7 122179547 IC50 = 5200 nM T94880 C1A0SQ 122179548 IC50 = 5000 nM T94880 C8KXV1 127025843 IC50 > 1000 nM T94880 CKS28E 127034802 IC50 = 71.9 nM T94880 C8ERJ7 127045762 IC50 > 1000 nM T94880 C7JC5K 134132904 IC50 = 25 nM T94880 C5DSV1 134134351 IC50 = 690 nM T94880 CYB46P 134135659 IC50 = 1300 nM T94880 CDH31O 134136945 IC50 = 13 nM T94880 C46XTD 134138113 IC50 = 940 nM T94880 CK75ZI 134138785 IC50 = 210 nM T94880 CCE1O4 134138988 IC50 = 31 nM T94880 C9V4CG 134140406 IC50 = 170 nM T94880 C5C4TS 134141052 IC50 = 1200 nM T94880 CWI41J 134141468 IC50 = 300 nM T94880 CYM06R 134142159 IC50 = 1200 nM T94880 CZB68J 134142873 IC50 = 78 nM T94880 CX03CP 134143856 IC50 = 1800 nM T94880 C5C2TA 134144975 IC50 = 94 nM T94880 CE12IN 134145489 IC50 = 1100 nM T94880 CM4U6L 134147181 IC50 = 54 nM T94880 CBES34 134147807 IC50 = 53 nM T94880 C60FLZ 134148014 IC50 = 38 nM T94880 CDUX09 134148124 IC50 = 2000 nM T94880 CGIT02 134149104 IC50 = 57 nM T94880 C4CA2M 134149641 IC50 = 110 nM T94880 C36GLZ 134150279 IC50 = 7.5 nM T94880 CZ42MI 134150952 IC50 = 190 nM T94880 C39AMZ 134151100 IC50 = 22 nM T94880 C10BFN 134151512 IC50 = 170 nM T94880 C8M3RH 134152780 IC50 = 44 nM T94880 C5PV8R 134153049 IC50 = 39 nM T94880 C4M7XF 134153576 IC50 = 170 nM T94880 C4AR9L 134153778 IC50 = 350 nM T94880 C6GC3U 134154700 IC50 = 130 nM T94880 C20PJY 134156194 IC50 = 60 nM T94880 CHN5R6 134156911 IC50 = 300 nM T94880 C70ZRI 134157187 IC50 = 49 nM T94880 C25ERN 137631967 IC50 > 1000 nM T94880 CI1E8V 137634241 IC50 > 10000 nM T94880 C06JRX 137637094 IC50 > 1000 nM T94880 C1DK0P 137651391 IC50 > 1000 nM T94880 CV5H3Z 137657932 IC50 > 1000 nM T94880 CE84NX 144944001 IC50 = 143 nM T94880 C65YWX 145964882 IC50 > 10000 nM T94880 CHC3T0 145965031 IC50 > 10000 nM T94880 CP92ZF 145965329 IC50 > 10000 nM T94880 C9HXI4 145966620 IC50 > 10000 nM T94880 CQE9M5 145966810 IC50 = 3670 nM T94880 C1EH6C 145967078 IC50 > 10000 nM T94880 CWJ12M 145969155 IC50 = 600 nM T94880 CGW5S1 145969844 IC50 > 10000 nM T94880 CB8R3A 145970271 IC50 > 10000 nM T94880 C40VIL 145972979 IC50 > 10000 nM T94880 CQBY19 145974023 IC50 = 1900 nM T94880 C4X7CT 145977420 IC50 > 10000 nM T94880 CLA57T 145978300 IC50 > 10000 nM T94880 C6KDQ5 145979093 IC50 = 268 nM T94880 CV7QY8 145981517 IC50 = 21 nM T94880 CG0R3A 145984368 IC50 = 690 nM T94880 CV78XO 145985621 IC50 = 445 nM T94880 CX5MB2 145986730 IC50 = 150 nM T94880 C1V6RA 145988134 IC50 > 100000 nM T94880 CD98JK 145989189 IC50 = 266 nM T94880 CWH69B 145989428 IC50 = 24 nM T94880 CZCS58 145989494 IC50 = 9 nM T94880 C0PHA7 145990595 IC50 = 4700 nM T94880 CN6T4K 145991513 IC50 = 270 nM T94880 CMBH76 145991936 IC50 = 27 nM T94880 C0SO4N 145993259 IC50 = 50 nM T94880 CI7F4G 145994227 IC50 = 11 nM T94880 C2MD1Q 155513187 IC50 > 10000 nM T94880 CTSM92 155538441 IC50 = 50 nM T94880 C40IYS 155562258 IC50 = 41.1 nM T94880 D0O6OH 71553154 IC50 = 0.7 nM T75015 D03HUX 49792852 IC50 > 10000 nM T75015 D0H9FR 118295624 IC50 = 792 nM T75015 D0O0LS 25141092 IC50 > 10000 nM T75015 D0RX8U 86281829 IC50 = 0.7943 nM T75015 CD8J9V 11963346 IC50 = 42 nM T75015 CS3EB6 16044861 IC50 = 37.9 nM T75015 C0Z6VU 16045086 IC50 = 4.1 nM T75015 CA1T2U 16045087 IC50 = 820 nM T75015 C35ILP 16045759 IC50 = 9100 nM T75015 CQ4O0Y 16045761 IC50 = 142 nM T75015 C1VS7Q 16045839 IC50 = 54 nM T75015 CCFT24 16046014 IC50 = 86.7 nM T75015 C6QT0J 44622837 IC50 > 1000 nM T75015 CU3RF1 45139989 IC50 > 10000 nM T75015 CQGZ06 45139991 IC50 > 10000 nM T75015 C7ON5A 46233287 IC50 > 10000 nM T75015 CF91RS 49843531 IC50 > 10000 nM T75015 CY48DE 49849970 IC50 = 31 nM T75015 C2Y6QS 50938552 IC50 > 10000 nM T75015 C36LQJ 50940491 IC50 = 1100 nM T75015 CWN54R 51003389 IC50 = 250 nM T75015 C9NYP4 51036677 IC50 > 10000 nM T75015 C4WRY3 51037112 IC50 > 10000 nM T75015 CRI28Z 51037948 IC50 > 10000 nM T75015 C3LTA4 53317522 IC50 = 6800 nM T75015 C87OAQ 53317986 IC50 = 140 nM T75015 CM0N2P 53319337 IC50 = 1300 nM T75015 C1L8WR 53319339 IC50 = 840 nM T75015 CC2IW7 53320600 IC50 = 1300 nM T75015 CN1TI4 53320630 IC50 = 7800 nM T75015 CZN0B8 53320631 IC50 = 300 nM T75015 C92UFO 53321929 IC50 = 102 nM T75015 CY0V2M 53323287 IC50 = 2500 nM T75015 C4HKE1 53323288 IC50 = 1600 nM T75015 CA4T3Y 53323289 IC50 = 4200 nM T75015 CNW02P 53323290 IC50 = 350 nM T75015 CP41WD 53324073 IC50 = 823 nM T75015 CJ4G3Y 53324074 IC50 = 3500 nM T75015 CL4G1V 53324616 IC50 = 5000 nM T75015 CNO54Z 53324617 IC50 = 442 nM T75015 C1EXW0 53325922 IC50 = 16 nM T75015 C2JB0Z 53325923 IC50 = 556 nM T75015 CD03BA 53466725 IC50 = 5.4 nM T75015 CXB94H 53466728 IC50 = 11.7 nM T75015 CYQ41S 53466951 IC50 = 1.3 nM T75015 C7QJ9O 53467174 IC50 = 1.9 nM T75015 CK7HG1 53467177 IC50 = 0.6 nM T75015 C5LS6O 53467178 IC50 = 0.2 nM T75015 CDU2A9 53467392 IC50 = 0.9 nM T75015 C3EYH5 53467617 IC50 = 2.5 nM T75015 CEU1I5 53467819 IC50 = 1.2 nM T75015 C1RMJ9 53467824 IC50 = 0.7 nM T75015 C09RAS 53468037 IC50 = 0.5 nM T75015 C37YIA 53468254 IC50 = 0.4 nM T75015 CYXW95 53468661 IC50 = 1.9 nM T75015 CCBA89 53468860 IC50 = 100 nM T75015 CX0R1K 53469059 IC50 = 30 nM T75015 CV7C0D 53469060 IC50 < 30 nM T75015 CCKD45 53469061 IC50 = 2.7 nM T75015 C91STB 53469449 IC50 = 0.2 nM T75015 CV6P9J 53469453 IC50 = 0.2 nM T75015 C8FS3Q 53469629 IC50 = 0.2 nM T75015 C56MKE 53469634 IC50 = 0.9 nM T75015 CZ1CI3 53469824 IC50 = 100 nM T75015 C7R2AX 66561010 IC50 = 7.4 nM T75015 CD52SV 66561011 IC50 = 8.1 nM T75015 C6SEL2 66561012 IC50 = 1.5 nM T75015 CCJ25F 66561013 IC50 = 17.4 nM T75015 C9Q0PT 66561090 IC50 = 0.2 nM T75015 CIXK72 66561167 IC50 = 0.3 nM T75015 CJD4Z1 66823478 IC50 = 0.5 nM T75015 CKOE90 71451677 IC50 = 11 nM T75015 CCN01X 71547862 IC50 > 10000 nM T75015 CW2YU7 72704111 IC50 = 19.1 nM T75015 CWCA98 72704112 IC50 = 23.4 nM T75015 CPIH57 72704113 IC50 = 63.8 nM T75015 CH1X8Y 72704114 IC50 = 57.5 nM T75015 CV39OD 72704115 IC50 = 16.6 nM T75015 CH63PM 86281830 IC50 = 12.59 nM T75015 CJ9U3A 86281960 IC50 = 3.162 nM T75015 CX4H6I 86583042 IC50 = 41 nM T75015 CVR43W 86583044 IC50 = 9 nM T75015 CA81UY 86583045 IC50 = 84 nM T75015 CY0UC4 90645194 IC50 > 10000 nM T75015 C8GWQ4 117636459 IC50 = 251.19 nM T75015 CKA4U9 117636465 IC50 = 10 nM T75015 C9IN8R 117636472 IC50 = 0.3981 nM T75015 CI5L3E 117636490 IC50 = 6.31 nM T75015 C7M9VF 117636502 IC50 = 1.585 nM T75015 CH9E1Q 117636508 IC50 = 5.012 nM T75015 CY7BI2 118706214 IC50 > 10000 nM T75015 CC6T5H 118720605 IC50 = 0.631 nM T75015 C5QC8E 118730408 IC50 = 1 nM T75015 C4TXF2 118730409 EC50 = 520 nM T75015 CN2A9O 118730410 IC50 = 3 nM T75015 COF69K 118730411 IC50 = 1 nM T75015 CEJ1S6 118730412 IC50 = 240 nM T75015 CQ0T5Z 118730413 IC50 = 140 nM T75015 CF47CO 118730414 EC50 = 130 nM T75015 CEJ67D 118730415 EC50 = 200 nM T75015 C5SI6Q 118730416 IC50 = 5 nM T75015 CR0H9D 118730417 IC50 = 240 nM T75015 CGDW48 118730418 EC50 = 190 nM T75015 C23KFD 118730419 IC50 = 11 nM T75015 CJ9SA8 118730420 IC50 = 53 nM T75015 C0HK5A 118730421 IC50 = 79 nM T75015 C1Q0UN 118730422 EC50 = 1300 nM T75015 C1K0PE 118730423 IC50 = 12 nM T75015 CHA4N2 136013680 IC50 > 10 nM T75015 C3COS8 136160805 IC50 = 18 nM T75015 C1YUD0 136219394 IC50 > 10 nM T75015 CIU8W3 136254389 IC50 > 10 nM T75015 C2MD1Q 155513187 IC50 > 10000 nM T75015 D08HFG 24809764 IC50 > 10000 nM T75015 D09HVH 135566652 IC50 > 10 nM T75015 D0N4LR 53469448 IC50 < 30 nM T82665 D05EAM 4735 IC50 = 582000 nM T82665 D0CR7L 90241742 IC50 = 6.2 nM T82665 C5P3TH 65130 IC50 = 357000 nM T82665 C0O3TQ 126437 IC50 = 166000 nM T82665 CRX9M1 725940 IC50 = 100 nM T82665 CQEF34 1002773 IC50 = 330 nM T82665 C8G4OE 1192043 IC50 = 14000 nM T82665 C69LIG 2850857 IC50 = 517 nM T82665 CCQ5K8 4720258 IC50 = 2800 nM T82665 C6OK4S 4973478 IC50 = 700 nM T82665 CH9K1U 5351747 IC50 = 712000 nM T82665 CW54YZ 9563572 IC50 = 570 nM T82665 CEKH37 10979651 IC50 = 186000 nM T82665 CH9JW4 40779692 IC50 = 1500 nM T82665 CPL71I 54596764 IC50 > 100000 nM T82665 CER5F1 67466175 IC50 > 100000 nM T82665 C5QE6A 67988955 IC50 > 50000 nM T82665 CAFU69 70686225 IC50 = 9100 nM T82665 CBK3U0 73892806 IC50 = 43000 nM T82665 C4XJ5N 78357767 IC50 > 100000 nM T82665 C10TUK 91667431 IC50 > 10000 nM T82665 CAO87S 91886006 IC50 = 109 nM T82665 C7G3KE 101982305 IC50 = 35 nM T82665 CG83ZK 118731732 IC50 = 1400 nM T82665 CWG18C 118731739 IC50 = 8360 nM T82665 CI1AE0 118731742 IC50 = 7040 nM T82665 C6Y8BM 118731746 IC50 = 35400 nM T82665 CV0FW8 121225442 IC50 = 2400 nM T82665 CIZF42 122178085 IC50 > 50000 nM T82665 CIOL82 122195095 IC50 > 100000 nM T82665 CSK94P 122497021 Ki = 0.02 nM T82665 CHO0M8 122497045 IC50 = 1 nM T82665 CIGD42 122669401 EC50 = 40 nM T82665 C6KV9H 124081151 IC50 > 100000 nM T82665 CSNE75 126637557 IC50 = 125 nM T82665 CHIO95 126637780 IC50 = 1070 nM T82665 C5Q4YV 126637809 IC50 = 0.25 nM T82665 CC48BQ 126638103 IC50 = 79.4 nM T82665 CT6K0X 126638123 IC50 = 0.4 nM T82665 CD5I8G 126638557 IC50 = 0.16 nM T82665 C1KH4F 126638569 IC50 = 51.3 nM T82665 CEG81V 126638570 IC50 = 7.9 nM T82665 CQWC72 130406427 IC50 = 26 nM T82665 CAT5Y8 132190219 IC50 = 1 nM T82665 CD72ZT 132190245 IC50 = 1 nM T82665 CIG7O9 132200399 IC50 = 1 nM T82665 CGQJ71 132200405 IC50 = 1 nM T82665 CD36BZ 132200436 IC50 = 1 nM T82665 C1Q9HM 132200647 IC50 = 1 nM T82665 C6WV9I 132200649 IC50 = 2 nM T82665 CJ0DK8 132200651 IC50 = 1 nM T82665 CYG96Q 132200704 IC50 = 1 nM T82665 C9YP3Z 132205208 IC50 = 2 nM T82665 C1UAJ8 134416883 IC50 = 6.31 nM T82665 CP5L9B 134416983 IC50 = 1.26 nM T82665 CDZ05F 134417152 IC50 = 6.31 nM T82665 CZ8OC0 135308090 IC50 > 1000 nM T82665 CY27NF 135308504 IC50 = 158 nM T82665 C7EC6X 135308815 IC50 > 1000 nM T82665 CQ0ZO4 135308826 IC50 = 12 nM T82665 CJMV78 135316976 IC50 = 43 nM T82665 CVW0C6 135318312 IC50 = 63 nM T82665 C4LK1X 137635057 IC50 > 50000 nM T82665 CRT8Q3 137655207 IC50 > 100000 nM T82665 CDPN65 137661881 IC50 > 50000 nM T82665 CV7MA4 138753159 IC50 = 22 nM T82665 CK2R6E 139449442 IC50 = 3.98 nM T82665 CV4YQ9 139449552 IC50 = 2 nM T82665 CTB83J 145983512 IC50 = 105 nM T82665 CK4ZT9 155175384 IC50 = 134 nM T82665 CD53BS 155520109 IC50 = 22 nM T82665 C1UAN2 155520348 IC50 > 500000 nM T82665 CN69BM 155523846 IC50 = 51 nM T82665 C7C8HI 155529624 IC50 > 30000 nM T82665 D00FLT 65482 IC50 = 8600 nM T82665 D02TVQ 71268957 IC50 > 100000 nM T82665 D05XQD 90241673 IC50 = 22 nM T82665 D09CLP 439155 IC50 = 200 nM T82665 D0L0DC 53339032 Ki = 1150 nM T02506 D00ZFP 5870 EC50 = 0.7 nM T02506 D01XBA 5035 Ki = 0.03 nM T02506 D06LOQ 179337 EC50 = 0.2 nM T02506 D06NXY 5991 IC50 = 2 nM T02506 D06XMU 6013 IC50 > 10000 nM T02506 D07BSQ 5994 IC50 > 1000 nM T02506 D07KSG 2733526 IC50 = 8 nM T02506 D08QMX 5757 EC50 = 0.004 nM T02506 D09NMD 216416 IC50 = 1.3 nM T02506 D0D1SG 5755 Ki > 5000 nM T02506 D0EP0C 5833 Ki > 1100 nM T02506 D0JO7Y 104741 IC50 = 0.06 nM T02506 D0JY8T 154257 IC50 = 3.7 nM T02506 D0Q4SD 443872 IC50 > 10000 nM T02506 D0V9BD 2375 Ki > 100000 nM T02506 D0X1EZ 2898 EC50 = 26 nM T02506 D0Y2NE 448537 EC50 = 0.007 nM T02506 D0Y7IU 5281004 IC50 > 10000 nM T02506 D0Y7JU 9854489 IC50 > 5000 nM T02506 D0Z1FX 5756 EC50 = 1.995 nM T02506 D0Z4EI 55245 Ki > 200 nM T02506 D00JFE 56941241 Ki = 0.37 nM T02506 D01SYU 10026128 IC50 = 10000 nM T02506 D07LZH 656954 IC50 = 1216 nM T02506 D09NST 449459 IC50 = 0.79 nM T02506 D0L4FS 5280961 IC50 = 9.7 nM T02506 D0LI1C 44469321 IC50 > 30000 nM T02506 D0R2SK 10286159 Ki = 2.29 nM T02506 D0SZ1G 121248172 IC50 > 100000 nM T02506 D0TN6K 118574930 IC50 = 6 nM T02506 D0U3EP 445154 Ki = 785 nM T02506 D0X1OW 86287635 IC50 = 0.138 nM T02506 D0X9YP 67041274 IC50 > 10000 nM T02506 D02KAU 46871935 IC50 > 10000 nM T02506 D03KTE 16750192 Ki > 10000 nM T02506 D05BCA 68570 EC50 = 1.5 nM T02506 D08DZZ 10634 EC50 = 26 nM T02506 D08HIH 6102691 IC50 = 210 nM T02506 D09AAM 104772 IC50 = 50 nM T02506 D09UFV 24825740 IC50 > 10000 nM T02506 D0H5CV 130936 IC50 = 25 nM T02506 D0J4ZH 3033898 Ki = 46.29 nM T02506 D0R8TB 6433099 EC50 = 0.1 nM T02506 D0U7OU 3220 Ki = 770 nM T02506 D0W5RL 9577221 IC50 = 1900 nM T02506 CXMH37 6620 IC50 = 133 nM T02506 C3EUZ1 6776 Ki = 310 nM T02506 C8GBH5 7184 IC50 = 1420 nM T02506 C6QYD8 8434 EC50 = 38200 nM T02506 CHA7C3 12111 EC50 = 909 nM T02506 CVUW13 14128 IC50 = 8970 nM T02506 CGWM38 54900 IC50 = 0.72 nM T02506 CSI62C 62082 EC50 = 6.5 nM T02506 CQ0IC4 63062 Ki = 0.04 nM T02506 CH98UA 65511 IC50 = 34600 nM T02506 CF5JU9 75386 IC50 = 230 nM T02506 CYCI69 80152 EC50 = 75.1 nM T02506 CNT0H1 96201 IC50 = 170 nM T02506 CS8Q6W 99649 Ki = 5700 nM T02506 CMEN50 101689 IC50 > 5000000 nM T02506 CM9CO5 119588 Ki = 41.5 nM T02506 C5E2IG 223998 Ki = 8 nM T02506 C78YGO 232446 IC50 = 520 nM T02506 C8MJB2 247310 IC50 = 84 nM T02506 CDHI70 251929 IC50 = 640 nM T02506 C9XC2A 252281 IC50 > 10000 nM T02506 CDP78A 261349 EC50 = 540 nM T02506 CZJW92 348148 EC50 = 80 nM T02506 C7HME8 439246 IC50 = 75302 nM T02506 CKB57V 440624 IC50 = 11000 nM T02506 C5SEF1 442342 IC50 1000000 nM T02506 C40YBS 444036 IC50 > 10000 nM T02506 CJZO27 445920 Ki = 4.1 nM T02506 CK01NI 448577 IC50 = 0.8 nM T02506 CGT37O 449205 IC50 = 0.5 nM T02506 C9AXQ3 449207 IC50 = 0.4 nM T02506 CBD7O2 449208 IC50 = 1.3 nM T02506 CL26SB 449209 IC50 = 1.3 nM T02506 CMT3P0 480764 EC50 = 5 nM T02506 C5UM8B 513197 EC50 = 1400 nM T02506 C0CF9H 586500 IC50 = 85700 nM T02506 CZ0AH3 638278 IC50 = 1870 nM T02506 C9UW8R 640096 EC50 = 2030 nM T02506 C2I3PM 646429 IC50 = 2230 nM T02506 CB20EC 656952 IC50 = 46 nM T02506 C67LKM 656953 IC50 = 1152 nM T02506 C2KCS3 667696 EC50 = 800 nM T02506 C2B0JA 674359 Ki = 15000 nM T02506 CX8H6W 687290 IC50 = 7980 nM T02506 C3R1PZ 721251 IC50 = 2320 nM T02506 C1OG7J 833976 EC50 = 12800 nM T02506 CV95AN 837745 IC50 = 28200 nM T02506 C31BFY 837746 EC50 = 31100 nM T02506 C69DLW 837838 IC50 = 4320 nM T02506 C4T6YS 837853 IC50 = 28100 nM T02506 C06JQG 837872 IC50 = 3060 nM T02506 CQOD41 837886 IC50 = 1000 nM T02506 C1ZE2H 845978 IC50 = 290 nM T02506 C6XGH8 849252 IC50 = 1200 nM T02506 C9S4EA 849257 IC50 = 2290 nM T02506 CE9VY2 849282 IC50 = 430 nM T02506 C4IQG9 849291 IC50 = 629 nM T02506 CN6RA2 849298 IC50 = 1980 nM T02506 CPQ72T 849308 IC50 = 31600 nM T02506 C45RBT 851153 EC50 = 3080 nM T02506 CO85AF 902564 EC50 > 100000 nM T02506 C5MZH8 906479 IC50 1000000 nM T02506 C2LRG9 927532 EC50 = 203 nM T02506 C5A7CD 928630 IC50 1000000 nM T02506 C90CUZ 1111980 EC50 > 10000 nM T02506 C6YNU8 1131384 Ki > 10000 nM T02506 C23KHO 1132609 IC50 < 100000 nM T02506 C5GJF1 1234611 IC50 = 3150 nM T02506 CM6NY1 1234663 IC50 = 1890 nM T02506 CMBE67 1234708 IC50 = 3290 nM T02506 C7TE0L 1717570 EC50 = 18700 nM T02506 CF4S1M 1731992 IC50 = 8770 nM T02506 C8WS4M 2040507 IC50 1000000 nM T02506 CLF0C9 2288503 IC50 = 24 nM T02506 CS6TF7 2733525 IC50 = 1700 nM T02506 C6LXG3 2747677 IC50 = 74 nM T02506 CFH19O 2887782 IC50 = 1100 nM T02506 CBZ6U1 3024714 IC50 = 285 nM T02506 C5GVH1 3035198 IC50 = 4 nM T02506 C7RNA9 3325226 IC50 = 16.48 nM T02506 C0F8EP 3519901 EC50 = 400 nM T02506 C9S2LO 4055843 EC50 = 4130 nM T02506 C6J0ZF 4369568 IC50 = 1.5 nM T02506 CFY94M 4369569 IC50 = 0.8 nM T02506 CL9G3U 4608762 EC50 > 10000 nM T02506 CH6RY7 5282240 EC50 = 11.2 nM T02506 CB6OK2 5287464 IC50 = 24 nM T02506 C7IBX9 5287551 IC50 = 8 nM T02506 CJB7T6 5288494 IC50 < 3.2 nM T02506 CW91XD 5322257 EC50 = 43.8 nM T02506 CS31LU 5322291 EC50 = 231 nM T02506 CP69KZ 5324349 EC50 = 21.4 nM T02506 C2JOL1 5327043 Ki = 0.47 nM T02506 CN7CS6 5372367 IC50 = 61.91 nM T02506 CF5VB6 5395460 IC50 1000000 nM T02506 C9GS2K 5397219 EC50 = 59.1 nM T02506 CQ83GI 5397398 IC50 1000000 nM T02506 C4Z1IB 5400235 EC50 = 331 nM T02506 CNG5W4 5407968 IC50 > 10000 nM T02506 CO36YU 5455071 EC50 = 35800 nM T02506 C52EHD 5822393 IC50 = 4660 nM T02506 CY9MR6 5885714 IC50 = 2320 nM T02506 CT0F6H 5948122 IC50 = 120 nM T02506 C6LCX3 6260040 EC50 = 415 nM T02506 CL41HW 6303362 EC50 = 95 nM T02506 C16ZSG 6439929 IC50 = 62000 nM T02506 C6RDY2 6444422 EC50 = 0.52 nM T02506 C3E0BP 6604873 EC50 = 2.9 nM T02506 C1VLY9 6918261 IC50 = 0.04 nM T02506 CF61LI 7314046 IC50 = 255 nM T02506 CM5Y0Z 7314049 IC50 = 795 nM T02506 CXHO01 7314090 IC50 = 10800 nM T02506 CFM7Q8 7314234 IC50 = 2870 nM T02506 C3M7RE 9804246 IC50 = 31 nM T02506 CU3QR8 9808162 Ki = 120 nM T02506 CNJE78 9811391 IC50 = 80 nM T02506 CE23GX 9814262 IC50 = 624 nM T02506 C34IZS 9814547 IC50 = 114 nM T02506 CZA2O0 9814673 EC50 = 794 nM T02506 CCUR98 9815144 IC50 = 344 nM T02506 CTB3F6 9815173 IC50 = 24 nM T02506 C4C7HN 9816479 IC50 > 200000 nM T02506 CNJK98 9816989 Ki = 10 nM T02506 CX1F7P 9819159 IC50 = 122.7 nM T02506 CTXR52 9820272 EC50 > 100000 nM T02506 CT78HP 9823190 IC50 > 10000 nM T02506 CN9M3P 9824019 Ki = 0.9 nM T02506 C94INP 9829162 IC50 = 2430 nM T02506 C7V2ZD 9835427 IC50 = 1650 nM T02506 CCX60E 9835779 IC50 = 1050 nM T02506 CHE70V 9838722 Ki > 100000 nM T02506 CS97CD 9846731 IC50 = 1 nM T02506 C2LV3C 9848252 IC50 = 1 nM T02506 CMI0N6 9848501 Ki = 0.32 nM T02506 CQGZ49 9856356 EC50 > 1000 nM T02506 CVW25C 9856632 EC50 = 671 nM T02506 C8ER6V 9869745 Ki = 210 nM T02506 C9MA0B 9878811 EC50 = 59 nM T02506 CIA6K1 9878841 EC50 = 460 nM T02506 CJ8VH6 9879228 IC50 = 5982 nM T02506 CPF25S 9879409 IC50 = 2420 nM T02506 CA1CJ6 9879798 IC50 = 273 nM T02506 C01ZFV 9882789 IC50 > 10000 nM T02506 CIT93X 9884138 IC50 = 141 nM T02506 CL8E7Z 9890509 IC50 = 0.7 nM T02506 CL7UB1 9900112 IC50 = 195 nM T02506 C3EQA8 9900383 EC50 = 449 nM T02506 C30BCU 9900479 IC50 = 264 nM T02506 CM9S2I 9900695 IC50 = 883 nM T02506 C3C6GN 9902151 IC50 = 41 nM T02506 C2BUL1 9902785 EC50 = 561 nM T02506 C38PGE 9903336 IC50 = 9.5 nM T02506 CB63ZP 9907598 IC50 = 500 nM T02506 CLC48G 9909681 IC50 = 0.5 nM T02506 CCZ9P8 9911175 Ki > 10000 nM T02506 CD3A6G 9912022 Ki = 0.6 nM T02506 C6YGM0 9912245 IC50 = 3 nM T02506 C58PVC 9921352 IC50 = 455 nM T02506 CJL2P9 9921784 IC50 = 976 nM T02506 CBX75P 9922298 IC50 = 30 nM T02506 CGN5C8 9922681 EC50 = 681 nM T02506 CX9AV7 9923647 EC50 = 1267 nM T02506 CJD4H0 9923941 IC50 = 70.5 nM T02506 CFT7M0 9924049 IC50 = 19 nM T02506 C9I3SQ 9924986 IC50 = 1410 nM T02506 CE6HU3 9925763 Ki = 4.34 nM T02506 CP8ZG3 9927355 Ki = 11 nM T02506 C39EXP 9933936 IC50 = 2281 nM T02506 CVW4Y8 9935633 IC50 = 7.8 nM T02506 CB0H3V 9942858 IC50 = 1210 nM T02506 CB65XA 9943599 IC50 > 10000 nM T02506 CW4RV2 9945087 EC50 = 1178 nM T02506 CO4IM2 9946131 IC50 = 663 nM T02506 C81CGQ 9946229 EC50 = 870 nM T02506 CZP05L 9948127 Ki = 3.3 nM T02506 CQ04ES 9948426 IC50 > 10000 nM T02506 CY6M2H 9953602 IC50 = 10.69 nM T02506 C9OPU4 9957008 Ki = 160 nM T02506 CEK90Y 9958368 Ki = 3.9 nM T02506 CO5V0P 9964601 IC50 = 1190 nM T02506 C0AJ3H 9964943 EC50 = 1233 nM T02506 CJT98P 9965271 IC50 = 630 nM T02506 C0LGC8 9965955 EC50 = 120 nM T02506 C1ZBV6 9967036 IC50 = 128 nM T02506 C29KIM 9968828 EC50 = 94 nM T02506 C4XGS5 9970588 Ki = 4 nM T02506 C05NAQ 9973567 IC50 = 597 nM T02506 CKS02X 9974556 EC50 = 620 nM T02506 COJ0E4 9993475 IC50 = 228 nM T02506 C4V6RF 9998996 IC50 > 1000 nM T02506 CB6AC7 10002045 IC50 = 1.4 nM T02506 CDU28H 10005346 IC50 = 2 nM T02506 CW4B6F 10015172 IC50 = 3074 nM T02506 CJN7T4 10016716 IC50 = 4160 nM T02506 C3XCR4 10016731 IC50 = 129 nM T02506 C7NLS3 10016946 IC50 = 7485 nM T02506 C8UT2P 10019713 IC50 = 4258 nM T02506 CG8B1H 10026593 IC50 = 1.6 nM T02506 CE0X1Y 10038212 IC50 = 1580 nM T02506 C0XGJ2 10043907 EC50 = 65 nM T02506 C3QBA5 10060912 IC50 = 14300 nM T02506 C9Z0AT 10060945 IC50 = 159 nM T02506 CUCM03 10062125 Ki > 100000 nM T02506 CIY1Z7 10064013 IC50 = 2521 nM T02506 C37ZQE 10072011 Ki = 8.69 nM T02506 C8P1BZ 10084254 IC50 = 3030 nM T02506 CDM8V3 10084479 IC50 = 716 nM T02506 CT1ZO9 10085265 IC50 = 33248 nM T02506 CYH2U5 10086047 IC50 = 627 nM T02506 CMDP60 10107798 IC50 > 10000 nM T02506 CM4B3Q 10108320 IC50 = 1160 nM T02506 C96JZH 10113416 IC50 = 4.7 nM T02506 C4XU7H 10115709 IC50 = 1 nM T02506 C9EDV6 10115710 IC50 = 0.8 nM T02506 CCA85G 10125282 IC50 = 55 nM T02506 CWLS93 10125319 IC50 = 1402 nM T02506 CTF5J0 10125414 Ki = 0.35 nM T02506 CH4N0B 10125582 IC50 = 356 nM T02506 CYIT90 10125667 IC50 = 10 nM T02506 CRP1U3 10128287 IC50 = 0.7 nM T02506 C08BYF 10140504 IC50 = 0.7 nM T02506 CQK5X9 10144672 Ki = 475 nM T02506 CC24WL 10149300 IC50 > 5000 nM T02506 CO1AE6 10149393 IC50 = 1650 nM T02506 C8G4PV 10149522 IC50 = 10 nM T02506 CY15UJ 10149610 IC50 = 118 nM T02506 C2EOX1 10151898 IC50 = 0.61 nM T02506 CIEH85 10154586 EC50 = 49 nM T02506 C0MX7K 10157532 IC50 > 10000 nM T02506 C1BAI4 10171529 Ki = 40 nM T02506 CT5W0A 10171640 IC50 = 12 nM T02506 CD36GZ 10171641 IC50 = 3.1 nM T02506 C36ACW 10171666 IC50 = 143 nM T02506 C5I7DH 10171723 Ki = 2.88 nM T02506 C9P4CF 10171732 IC50 = 548 nM T02506 C5DSH0 10171830 IC50 = 125 nM T02506 C3QR7A 10171898 IC50 = 9 nM T02506 CK0ZU9 10172081 IC50 = 710 nM T02506 C1VDO4 10174471 IC50 = 3.8 nM T02506 CJO0M8 10174620 IC50 = 1.1 nM T02506 C2YRA6 10177915 IC50 = 124 nM T02506 C8L7HJ 10179031 IC50 > 10000 nM T02506 C2BS8L 10181886 Ki = 1.7 nM T02506 CWCM45 10182934 Ki = 0.6 nM T02506 C3JZH5 10183377 EC50 = 200 nM T02506 CKT6Z4 10183386 IC50 = 18 nM T02506 CQB51M 10184149 IC50 = 0.9 nM T02506 C0J9AT 10184212 IC50 = 5.2 nM T02506 CG5N8H 10184413 Ki = 490 nM T02506 C8XEP4 10192873 IC50 = 180 nM T02506 CR48FY 10192874 IC50 > 5000 nM T02506 CP70BT 10192899 IC50 = 21 nM T02506 C3RV4A 10192967 Ki = 41 nM T02506 CT19KI 10192968 Ki = 65 nM T02506 CVM71O 10192978 IC50 = 1056 nM T02506 CY3ZU9 10193027 IC50 = 114 nM T02506 C1UF6W 10193573 IC50 = 200 nM T02506 C73GTR 10204098 IC50 = 11.9 nM T02506 CS91YM 10210142 Ki = 675 nM T02506 CH02FU 10214626 IC50 = 6 nM T02506 C4PKF0 10214678 Ki = 267 nM T02506 CJN2Y4 10214684 IC50 > 5000 nM T02506 CP90ZM 10214912 IC50 = 480 nM T02506 C82SVD 10215058 IC50 = 299 nM T02506 C8GZN0 10215089 IC50 = 5.2 nM T02506 CP4U5C 10215240 IC50 = 47 nM T02506 CP41MR 10215241 IC50 = 3 nM T02506 C7PSG6 10215290 IC50 = 21 nM T02506 C0FU1V 10215342 IC50 = 131 nM T02506 CP1S2V 10217796 IC50 = 4 nM T02506 CU2RI4 10217951 IC50 = 1 nM T02506 CW05OU 10218853 IC50 > 10000 nM T02506 CJ9BE0 10222329 IC50 > 10000 nM T02506 C84SRT 10223610 IC50 > 10000 nM T02506 CGF4E7 10226687 IC50 = 3 nM T02506 C7FXG9 10227720 IC50 = 172 nM T02506 C5M1RH 10229852 Ki = 360 nM T02506 CNB84J 10236378 IC50 = 2951 nM T02506 CVMD95 10236407 IC50 = 58 nM T02506 CV9SZ3 10236450 IC50 = 109 nM T02506 C1K8OP 10236507 IC50 = 2 nM T02506 C7CPB9 10238739 IC50 = 51 nM T02506 CMY87N 10243978 EC50 = 6.7 nM T02506 C7E0OP 10244111 IC50 = 488 nM T02506 C0JE2W 10248828 IC50 = 1440 nM T02506 CJQZ83 10254189 Ki = 0.5 nM T02506 CS4B5C 10265236 IC50 = 46 nM T02506 CPBH94 10266789 IC50 = 43 nM T02506 CGV0O2 10268080 IC50 = 196 nM T02506 CR59SC 10271193 IC50 > 10000 nM T02506 CPIS57 10271557 IC50 > 10000 nM T02506 CPZY03 10275313 Ki = 2.5 nM T02506 C7LHP1 10275916 Ki > 1000 nM T02506 CL5P3T 10276036 Ki = 120 nM T02506 CBD8V6 10282029 EC50 = 150 nM T02506 C7G4RE 10286186 IC50 = 40 nM T02506 C15UPR 10286213 IC50 = 40 nM T02506 C37GHD 10286369 IC50 = 35 nM T02506 C4U9ZV 10286370 IC50 = 519 nM T02506 CS4Y7Z 10286462 IC50 = 290 nM T02506 CUQC81 10287415 IC50 > 1000 nM T02506 CM8IW0 10288944 IC50 = 2.6 nM T02506 CLOE40 10291224 IC50 = 5880 nM T02506 C04JEC 10299557 IC50 = 110 nM T02506 C10CJA 10308134 IC50 = 105 nM T02506 CGR20A 10308169 IC50 = 31 nM T02506 C1KY6P 10308176 IC50 = 23 nM T02506 CX15KH 10308458 IC50 = 36 nM T02506 C7R4NE 10308501 Ki = 6.11 nM T02506 C0VUR6 10308538 IC50 = 580 nM T02506 COP14A 10312439 IC50 > 1000 nM T02506 COHA43 10316618 IC50 = 225 nM T02506 C1FLQ0 10323601 Ki = 34 nM T02506 CPJS68 10324755 Ki = 1.22 nM T02506 C5K2CL 10332429 IC50 > 10000 nM T02506 C7R6EP 10332721 IC50 = 1280 nM T02506 CO2IH4 10334049 IC50 = 4382 nM T02506 CPK7W1 10344612 Ki = 32 nM T02506 C0YAJ6 10344970 IC50 = 0.7 nM T02506 CEA16J 10344977 IC50 = 2.7 nM T02506 C1MH2K 10346077 EC50 = 1800 nM T02506 C35BTN 10355544 IC50 = 10000 nM T02506 CMY0N8 10355768 IC50 = 435 nM T02506 C61WZX 10356510 IC50 = 9830 nM T02506 C5YU0I 10358550 IC50 = 6850 nM T02506 CR98BH 10358677 IC50 = 1920 nM T02506 C7SO6W 10361788 IC50 = 9 nM T02506 CEJ78I 10365592 IC50 > 2000 nM T02506 CKD8I0 10370518 IC50 = 5 nM T02506 CBG59N 10377168 IC50 = 550 nM T02506 CGCE89 10378417 IC50 = 484 nM T02506 CRB41T 10379126 IC50 = 25956 nM T02506 C14AIB 10384345 IC50 > 2000 nM T02506 C6RQK1 10386584 IC50 > 10000 nM T02506 CYN9E1 10390108 EC50 = 200 nM T02506 CK8MI6 10390296 IC50 = 1.3 nM T02506 CH9P0A 10390835 IC50 = 61 nM T02506 CJV0O5 10400919 IC50 = 1780 nM T02506 C7JN6F 10401620 IC50 = 626 nM T02506 C40NPC 10407651 Ki > 100000 nM T02506 CQ46GH 10412249 Ki = 0.28 nM T02506 C1P4XA 10414598 IC50 = 5.6 nM T02506 CA80YJ 10423234 IC50 = 11097 nM T02506 C6H7EJ 10423780 IC50 = 10000 nM T02506 CPM1L8 10425817 IC50 = 11600 nM T02506 CC1V4Y 10428321 IC50 = 373 nM T02506 C98YGB 10430074 IC50 = 597 nM T02506 C04EKD 10436416 IC50 > 10000 nM T02506 C8ZS3V 10447061 IC50 > 6260 nM T02506 CZ08NR 10447944 IC50 = 29.8 nM T02506 CH58OG 10450569 EC50 = 15 nM T02506 C0NT9D 10454007 IC50 > 5000 nM T02506 CM92LK 10467580 IC50 = 583 nM T02506 C4JK0T 10468337 IC50 = 785 nM T02506 CLV49C 10470279 EC50 = 243 nM T02506 C6UMY7 10471178 IC50 = 3120 nM T02506 CB8PK9 10473796 EC50 = 1740 nM T02506 C85RBN 10474264 IC50 > 2000 nM T02506 CUL8O4 10475384 IC50 > 1000 nM T02506 CMG35I 10478373 IC50 = 2.5 nM T02506 C8GZN6 10479379 IC50 = 1.9 nM T02506 CZB0G1 10480448 IC50 = 65 nM T02506 CAL8E3 10719917 IC50 = 0.046 nM T02506 CM69RP 10768122 Ki = 0.25 nM T02506 CC7N5G 10809406 IC50 > 11 nM T02506 C30MWO 10812923 EC50 = 1660 nM T02506 CC2L7D 10814352 IC50 < 0.002 nM T02506 C39FWK 10858337 EC50 = 40 nM T02506 CKTE95 10863480 Ki > 10000 nM T02506 CT1L6K 10874604 Ki > 10000 nM T02506 C2W9QX 10885394 IC50 = 71 nM T02506 C75IVW 10892270 EC50 = 464 nM T02506 C4ZI0B 10897174 Ki > 10000 nM T02506 CNZ9H2 10901682 EC50 = 191 nM T02506 CMW1U8 10906531 Ki = 1420 nM T02506 CJP54O 10906754 Ki = 200 nM T02506 CY5R8D 10908233 Ki = 1050 nM T02506 C40LHE 10917513 Ki > 10000 nM T02506 C3WI4P 10917876 IC50 = 46 nM T02506 CJ8OD1 10923143 EC50 = 18 nM T02506 CU46XG 10928571 IC50 = 2.9 nM T02506 CS24AP 10928882 IC50 = 3.097 nM T02506 COM46T 10929139 Ki = 145 nM T02506 CJ3RF6 10930298 Ki = 1300 nM T02506 C3HG2S 10933614 EC50 = 178 nM T02506 C5E8VA 10938971 Ki = 5130 nM T02506 CK5D4I 10939453 IC50 = 0.6998 nM T02506 CT8B7X 10940598 Ki = 180 nM T02506 C1OQB3 10945098 EC50 = 71200 nM T02506 CH14AY 10950078 Ki = 6870 nM T02506 CJL36T 10950356 Ki > 10000 nM T02506 CZ8F4V 10950649 IC50 = 2.897 nM T02506 CP2IK4 10950883 IC50 = 4.498 nM T02506 C3I5PB 10952341 Ki = 1450 nM T02506 C4VD3H 10955612 EC50 = 3.1 nM T02506 CR94QD 10956181 EC50 = 148 nM T02506 CD90TL 10961334 Ki = 2400 nM T02506 CZGP46 10967017 EC50 = 16 nM T02506 CI9PC0 10972569 EC50 = 500 nM T02506 C7KSR9 10972765 Ki = 570 nM T02506 CW7ND8 10973721 Ki = 6320 nM T02506 CW52ES 10973841 Ki = 810 nM T02506 CC4UT6 10978897 EC50 = 2.9 nM T02506 C93KBD 10978965 EC50 > 1000 nM T02506 CF2WJ3 10983822 Ki = 560 nM T02506 C2Q9UC 10985075 Ki = 855 nM T02506 C79JBL 10993930 IC50 = 2.6 nM T02506 CL1I0Z 10994057 Ki = 290 nM T02506 CW62AM 10999188 EC50 = 269 nM T02506 C1N8ZM 10999677 EC50 = 48 nM T02506 CGSE70 11011115 EC50 = 2.7 nM T02506 CE4C5I 11015765 IC50 = 2.999 nM T02506 CWO8S9 11016369 Ki = 1000 nM T02506 CHR7A9 11016735 Ki = 125 nM T02506 CG37VC 11022432 EC50 = 162 nM T02506 CH9Y1B 11026647 IC50 = 0.5998 nM T02506 CGX1N0 11028495 Ki = 1130 nM T02506 COE9W8 11037182 Ki = 2370 nM T02506 CZW72E 11037591 IC50 = 3.5 nM T02506 C3JH4N 11039284 Ki = 2040 nM T02506 CNG30Q 11048590 Ki > 10000 nM T02506 C2Z6TH 11048839 Ki = 415 nM T02506 CQN16G 11048858 IC50 = 3.3 nM T02506 C5W9IK 11060085 Ki = 2275 nM T02506 CWO84P 11060104 Ki = 830 nM T02506 CV1A6F 11070590 Ki = 1140 nM T02506 CF9LM6 11070635 Ki = 270 nM T02506 CU9PY6 11071460 EC50 = 180 nM T02506 CWG41U 11075979 EC50 = 23 nM T02506 C2L7DT 11086416 EC50 = 363 nM T02506 C09ZLY 11088436 Ki > 10000 nM T02506 CG3VQ7 11091722 IC50 = 1.5 nM T02506 C8ED0O 11092497 Ki = 480 nM T02506 C49GHR 11097061 EC50 = 0.38 nM T02506 CX8YU9 11102748 IC50 = 44 nM T02506 CD1G4U 11102972 Ki = 570 nM T02506 CR8OQ5 11114635 Ki = 2360 nM T02506 CDJW25 11117751 EC50 = 209 nM T02506 C1O8RD 11124781 Ki > 10000 nM T02506 CGH0S4 11135858 Ki = 570 nM T02506 CNEX86 11146178 Ki = 3000 nM T02506 CIG8Z6 11153316 Ki > 100000 nM T02506 CJ4S8B 11153461 EC50 > 10000 nM T02506 CJ12UZ 11155391 IC50 = 0.66 nM T02506 CS2B4Z 11155392 IC50 = 1.4 nM T02506 CJ7KZ9 11155655 Ki > 100000 nM T02506 CP7R9U 11156432 EC50 = 1700 nM T02506 C4SEB7 11160528 IC50 = 790 nM T02506 CGI4Y2 11162677 Ki > 1000 nM T02506 CT0JD9 11164713 EC50 > 1000 nM T02506 C5DM4H 11165305 IC50 = 38 nM T02506 C68FNC 11167858 IC50 = 1090 nM T02506 CX91QE 11185437 IC50 = 343 nM T02506 CVAI71 11186162 EC50 = 1000 nM T02506 CBS6E8 11197092 IC50 = 180 nM T02506 CAPL61 11197251 IC50 = 45 nM T02506 C9T6KS 11197891 Ki > 100000 nM T02506 CLQ9C4 11197931 Ki = 8.3 nM T02506 C1XPD4 11201600 IC50 = 18 nM T02506 CB1FI6 11201991 IC50 = 1.3 nM T02506 CO2N4Z 11208222 Ki > 100000 nM T02506 C0M4IP 11208678 Ki = 700 nM T02506 CN6V7O 11209303 Ki > 100000 nM T02506 CDG4Q2 11221797 EC50 > 10000 nM T02506 C3M5WN 11224950 IC50 = 2.4 nM T02506 CA7F5T 11225110 EC50 = 1500 nM T02506 C7M9AJ 11230651 Ki > 100000 nM T02506 CN27ZJ 11231364 IC50 = 73 nM T02506 C2Q5PJ 11231792 IC50 = 186 nM T02506 CMIO31 11235808 EC50 = 780 nM T02506 CQHW46 11243890 Ki > 100000 nM T02506 C3B4HX 11244016 Ki > 100000 nM T02506 C5IM4X 11247367 Ki = 1.7 nM T02506 C3RM9N 11254549 IC50 = 235 nM T02506 C5A7JR 11254851 IC50 = 406 nM T02506 CNJ4Q3 11255230 IC50 = 6324 nM T02506 CYCR06 11256303 IC50 > 10000 nM T02506 CWF3M2 11256602 Ki = 12.4 nM T02506 CEA6U1 11259746 IC50 = 5.1 nM T02506 CZ1LG3 11266077 Ki > 100000 nM T02506 CIRO56 11267448 IC50 = 64908.26 nM T02506 C7N9EL 11268331 IC50 = 116 nM T02506 CC0XI4 11279959 IC50 > 10000 nM T02506 C4SC0W 11281576 IC50 > 1000 nM T02506 C8LFT9 11287739 Ki > 100000 nM T02506 C69KHE 11294796 IC50 = 2.5 nM T02506 C5A1NL 11300439 IC50 = 96 nM T02506 CY2GB4 11300595 Ki = 380.8 nM T02506 CS5HC9 11300885 EC50 = 11 nM T02506 CI7CZ3 11301461 IC50 = 55 nM T02506 C0XUF2 11305564 IC50 > 5000 nM T02506 CP61NH 11310856 Ki > 100000 nM T02506 C8S5AR 11314096 Ki = 7.2 nM T02506 C5M2KX 11317852 IC50 = 0.7 nM T02506 COU8G6 11323885 IC50 = 434 nM T02506 C61YIJ 11326213 EC50 = 5000 nM T02506 C1HZS7 11336351 IC50 > 10000 nM T02506 CL0TH7 11338484 EC50 = 3470 nM T02506 C1ZJ2R 11338969 IC50 = 31 nM T02506 CH12WB 11339036 IC50 = 153 nM T02506 CT9Y4O 11339440 IC50 > 10000 nM T02506 CBN46V 11340868 Ki = 1.03 nM T02506 C2T7ZW 11350120 EC50 > 10000 nM T02506 CU6BE2 11350495 IC50 = 34.9 nM T02506 C6YUB4 11350836 IC50 = 38 nM T02506 CR1EB4 11351870 IC50 = 19.6 nM T02506 CSNT72 11357451 IC50 = 84 nM T02506 CW3L1T 11358876 Ki > 100000 nM T02506 C8Z3YW 11359856 Ki = 4.2 nM T02506 CT3WZ0 11361524 IC50 = 46.6 nM T02506 C8AW4J 11363477 IC50 = 1.3 nM T02506 C90MRZ 11368962 EC50 = 35 nM T02506 C1HS3D 11369558 IC50 = 113 nM T02506 CMSU02 11370317 Ki = 410 nM T02506 C68GMX 11375318 EC50 = 1820 nM T02506 CXO72T 11376166 EC50 = 85 nM T02506 CTL6Z7 11382252 EC50 = 3000 nM T02506 CEI5V6 11385564 IC50 = 119 nM T02506 CK42BA 11391793 IC50 = 247 nM T02506 CL8JI2 11391816 Ki > 100000 nM T02506 C8G2ED 11397112 IC50 = 1.6 nM T02506 C17SXG 11397412 IC50 = 0.5 nM T02506 CO15AK 11403179 IC50 = 73 nM T02506 CS6VA1 11406904 IC50 = 55 nM T02506 CUC6L8 11407390 IC50 = 87 nM T02506 C0L2IW 11414230 Ki > 100000 nM T02506 CYM9V2 11414783 Ki > 100000 nM T02506 CO20QH 11416730 IC50 > 10000 nM T02506 C9YW0P 11425113 Ki > 100000 nM T02506 CC9D7U 11427021 EC50 = 984 nM T02506 C5WO0U 11429662 IC50 > 1000 nM T02506 CM9VH4 11430588 IC50 = 63 nM T02506 CFXR09 11431084 EC50 = 500 nM T02506 CGF15N 11431657 IC50 = 177 nM T02506 C0VR7F 11437418 IC50 = 26 nM T02506 CP7J9V 11437506 IC50 = 231 nM T02506 CYIU98 11438491 Ki > 100000 nM T02506 C6QK5H 11441393 EC50 > 10000 nM T02506 C2NMY6 11465422 IC50 = 3 nM T02506 CFG6L2 11471499 IC50 = 527 nM T02506 C8B9ZT 11471500 IC50 = 254 nM T02506 CK75PT 11476995 IC50 = 2.84 nM T02506 CP4M8J 11482995 Ki = 136 nM T02506 CNUG46 11487991 IC50 = 1.5 nM T02506 C3PNE7 11493187 IC50 = 11111 nM T02506 C7D5BU 11493338 IC50 = 5365 nM T02506 CN3W8L 11493379 IC50 = 6200 nM T02506 CFPW12 11496802 Ki = 0.3 nM T02506 CM76FT 11496925 Ki = 1.89 nM T02506 CQZ37A 11515143 IC50 = 81324 nM T02506 C4OBS2 11517134 Ki = 692 nM T02506 C5W9CK 11517889 IC50 = 3.5 nM T02506 CJ2WY6 11522286 EC50 = 4.3 nM T02506 C9G5AE 11536973 EC50 = 494 nM T02506 C5W8HY 11537063 EC50 = 622 nM T02506 CMOL82 11540768 Ki = 0.57 nM T02506 CS0O5B 11554672 EC50 = 3100 nM T02506 CUK47O 11558075 IC50 = 15521 nM T02506 CWCZ35 11558237 IC50 = 13240 nM T02506 CR4D8K 11558528 EC50 = 982 nM T02506 CP9GR8 11561520 Ki = 2 nM T02506 CSF3D4 11565065 EC50 = 10600 nM T02506 CUD60X 11565235 IC50 = 9635 nM T02506 C5YO1V 11565733 IC50 = 55015 nM T02506 C7UDF3 11565847 IC50 = 10649 nM T02506 C19NWZ 11565922 EC50 = 344 nM T02506 CWOZ42 11572578 IC50 = 66860 nM T02506 C07ALM 11582925 IC50 = 14 nM T02506 CKV64Z 11582975 Ki = 28 nM T02506 C4IZK8 11587711 EC50 = 14 nM T02506 CGQ5M2 11587774 IC50 = 770 nM T02506 C29NKX 11597321 IC50 = 18000 nM T02506 C9QS7V 11605525 Ki = 5.8 nM T02506 C92NWX 11610210 IC50 = 5 nM T02506 CC21VD 11610867 Ki = 59 nM T02506 CNP72K 11615788 EC50 = 0.31 nM T02506 CA3ID6 11619024 Ki = 52 nM T02506 CB10RY 11623915 EC50 = 324 nM T02506 C8M6GX 11631082 EC50 = 47 nM T02506 C7PG3I 11633183 Ki = 60 nM T02506 C45XNL 11637913 IC50 = 43968 nM T02506 CQ8EI7 11638242 Ki = 0.67 nM T02506 C60DQS 11638602 EC50 = 603 nM T02506 CA7S2I 11644884 IC50 = 34626 nM T02506 C2MQE5 11644885 IC50 = 121 nM T02506 CD2TL1 11645057 EC50 = 158 nM T02506 C7NBT6 11645733 EC50 > 1000 nM T02506 CK7ZQ8 11647673 IC50 = 0.6 nM T02506 C9LZ1F 11651922 IC50 = 43814 nM T02506 C84GDU 11655056 IC50 = 13000 nM T02506 CI1E3R 11659178 EC50 = 0.059 nM T02506 C3GXI8 11659260 IC50 = 44175 nM T02506 C1QV8H 11660523 Ki = 198 nM T02506 CWL7S9 11662094 IC50 = 29000 nM T02506 C0LKN3 11663272 EC50 = 152 nM T02506 CF4HM7 11666535 IC50 = 19437 nM T02506 CX2W9Z 11666644 IC50 = 6247 nM T02506 CJ2UC4 11674336 IC50 = 101544 nM T02506 CB1DU8 11674420 EC50 = 17 nM T02506 C3IK0P 11680776 IC50 = 15297 nM T02506 CH7O4Y 11681405 IC50 = 178 nM T02506 CJL8A6 11681415 EC50 = 10 nM T02506 CFZ0K5 11688293 EC50 = 3.9 nM T02506 CZ35CY 11694886 IC50 = 70277 nM T02506 CQ0IP3 11695307 IC50 = 70399 nM T02506 C20PTC 11696330 Ki = 2.1 nM T02506 CC6VK8 11702683 EC50 = 719 nM T02506 C0FEB7 11710790 EC50 = 427 nM T02506 CG4E2O 11719093 Ki = 4 nM T02506 C43LND 11720175 Ki = 0.24 nM T02506 CRP5H6 11720774 EC50 = 100 nM T02506 CR52IJ 11722356 EC50 > 1000 nM T02506 C7D9HG 11724363 IC50 > 10000 nM T02506 CO3S2Z 11724477 IC50 = 10000 nM T02506 CWK56G 11730419 Ki = 1000 nM T02506 CBMR23 11730420 Ki > 10000 nM T02506 C4FXP3 11730578 Ki = 200 nM T02506 C4GDB9 11730602 IC50 = 5.2 nM T02506 CB8J4L 11730916 Ki = 60 nM T02506 C1I0ZW 11733031 Ki = 3240 nM T02506 CT40UX 11734564 Ki = 1025 nM T02506 CGZ40Y 11738040 IC50 = 312 nM T02506 C4DCI8 11738269 IC50 = 2329 nM T02506 C9I3LZ 11738605 EC50 = 344 nM T02506 CF0D1S 11740374 EC50 = 1860 nM T02506 CCT71E 11743602 Ki = 1380 nM T02506 C9KTN0 11744183 Ki = 1.1 nM T02506 C0K4LB 11749762 Ki = 49000 nM T02506 CEC20W 11750375 IC50 = 18.2 nM T02506 C5YF3X 11750707 IC50 = 162 nM T02506 C5JH1M 11751440 IC50 = 122 nM T02506 CA2DO6 11770898 IC50 = 98 nM T02506 CHX6E0 11776977 IC50 = 4590 nM T02506 CH7VT9 11777076 IC50 = 3710 nM T02506 CD4W6C 11777154 IC50 = 1860 nM T02506 C98FDE 11777375 EC50 = 138 nM T02506 CNLQ34 11777905 IC50 = 1000 nM T02506 CT8OB2 11777956 IC50 = 97982 nM T02506 CL76UG 11778912 EC50 > 1000 nM T02506 CS9K7Z 11812018 IC50 = 1.799 nM T02506 CS4X7T 11817441 Ki > 100000 nM T02506 C8YD5R 11823753 EC50 = 42 nM T02506 CYQ0W7 11826815 IC50 = 19 nM T02506 CUVE20 11826959 Ki = 680 nM T02506 CT6Z4P 11827881 Ki = 250 nM T02506 C2VDT9 11954121 IC50 = 5.9 nM T02506 CFB48H 11957006 IC50 = 793 nM T02506 C3F6JK 11977778 EC50 = 870 nM T02506 C2CXT4 11987846 IC50 = 129 nM T02506 CSK1Q4 12019124 IC50 > 5000 nM T02506 COR2Z7 12074176 Ki = 0.21 nM T02506 C2HNA8 12083341 IC50 = 2728 nM T02506 C4U8KY 12085089 IC50 > 10000 nM T02506 COZ0Q5 12085941 IC50 = 28.7 nM T02506 C0P4TJ 12085942 IC50 = 562 nM T02506 C06AOU 12117259 EC50 = 65 nM T02506 C0IJ4C 12130940 EC50 = 300 nM T02506 CD2K0P 12130943 EC50 = 150 nM T02506 C41TJX 12258274 IC50 = 3672 nM T02506 CTZ92I 12642771 IC50 = 39400 nM T02506 C5GV6L 13613337 IC50 = 2530 nM T02506 C1J0CU 13720325 EC50 = 4 nM T02506 CS38YQ 14065243 EC50 = 15 nM T02506 CK2O7U 14128123 EC50 = 1500 nM T02506 CTU56S 14496018 EC50 = 1200 nM T02506 C42MYO 15429026 IC50 = 10.9 nM T02506 CB7K0N 15521393 IC50 = 3.53 nM T02506 C9NSQ7 15542995 EC50 = 5 nM T02506 C9IUR6 15543000 IC50 = 94 nM T02506 C0Q5RP 15543001 EC50 = 13 nM T02506 CF0U2J 15543006 EC50 = 336 nM T02506 COW27A 15543007 EC50 = 28 nM T02506 CZB7P9 15543008 EC50 = 40 nM T02506 C8J6DM 15543009 IC50 = 3.5 nM T02506 C49NDP 15887827 EC50 = 10 nM T02506 CUO82C 15984114 EC50 = 10.4 nM T02506 C2CVH9 15984115 EC50 = 8.3 nM T02506 CWF0I6 16007239 EC50 = 519 nM T02506 CR2Q9N 16038396 Ki = 1700 nM T02506 CV4LD2 16082545 IC50 = 82 nM T02506 C7S4XY 16082546 IC50 = 440 nM T02506 CKGI59 16082547 IC50 = 5500 nM T02506 C5ZJR4 16082550 IC50 = 1200 nM T02506 CR8NQ7 16082556 IC50 = 22 nM T02506 CUOE19 16082557 EC50 = 14 nM T02506 CIWO01 16082558 EC50 = 11 nM T02506 CW2EC8 16082559 IC50 = 40 nM T02506 CZ3N1E 16082564 IC50 = 160 nM T02506 C9WS2L 16082565 IC50 = 140 nM T02506 COR9P3 16082566 EC50 = 300 nM T02506 CH8A7C 16082568 IC50 = 340 nM T02506 C9O5EM 16082572 IC50 = 14 nM T02506 CK7PI6 16082573 IC50 = 25 nM T02506 C9QXI4 16082574 IC50 = 25 nM T02506 C7GL5X 16082575 EC50 = 41 nM T02506 C2BOE6 16103238 Ki = 266 nM T02506 C4UFW5 16103245 Ki = 408 nM T02506 CKHS18 16106496 IC50 < 100000 nM T02506 C95OTV 16106497 IC50 < 100000 nM T02506 CT17EJ 16106503 IC50 < 100000 nM T02506 C6H0EQ 16655080 IC50 = 36 nM T02506 C1UY8J 16666386 IC50 > 5000 nM T02506 C1F5XE 16719760 IC50 = 666 nM T02506 CE6FQ8 16719863 IC50 = 35.6 nM T02506 C7N4LJ 16719865 Ki = 0.63 nM T02506 C0PMA8 16719866 IC50 = 19.3 nM T02506 CC82UX 16720250 IC50 = 27 nM T02506 CWK35C 16730429 IC50 = 29000 nM T02506 CM4BS9 16739367 IC50 = 2 nM T02506 CZ34MS 16750039 IC50 = 8 nM T02506 CVSA61 16750040 IC50 = 1 nM T02506 CQZK05 16758226 Ki = 43.8 nM T02506 C3M8BI 17010631 IC50 < 100000 nM T02506 CVBN30 17191222 IC50 = 44.43 nM T02506 CE4CP2 17756206 IC50 = 193 nM T02506 C2AP6N 17760561 EC50 = 2.6 nM T02506 C4DV6C 17964485 Ki = 88 nM T02506 C9B3MR 17972677 IC50 = 1990 nM T02506 C4UG6E 17972712 IC50 = 4410 nM T02506 C84OYE 18172398 IC50 = 4.7 nM T02506 CS1C5Q 18172400 IC50 = 30.7 nM T02506 C30ALH 18172403 IC50 = 165 nM T02506 CZ0VW4 18172409 IC50 = 385 nM T02506 C5U1YK 18172442 IC50 = 29.4 nM T02506 CJ05MC 18172444 IC50 = 42.7 nM T02506 CUS3Z9 18172448 IC50 = 160 nM T02506 C3X1FG 18172450 IC50 = 28 nM T02506 CTVK47 18172466 IC50 = 6.7 nM T02506 CR53UZ 18172469 IC50 = 24.8 nM T02506 C93MVX 18172476 IC50 = 9.2 nM T02506 CCE1L5 18172477 IC50 = 50 nM T02506 C0RZB8 18172482 IC50 = 235 nM T02506 C9DS4J 18695694 Ki = 2 nM T02506 CJ9RH8 19087421 IC50 > 200000 nM T02506 CGP29U 19793984 IC50 = 2900 nM T02506 C1F4KI 19793985 IC50 = 84 nM T02506 C95KIE 20160413 IC50 = 1.3 nM T02506 CI0P6T 20161167 IC50 = 14 nM T02506 CSY05K 20227298 IC50 = 1.3 nM T02506 CM86ZJ 20734982 IC50 = 3 nM T02506 C0Q4FT 21051956 IC50 = 0.28 nM T02506 CF0S6J 21210483 IC50 > 30000 nM T02506 CV2N4Y 21252247 EC50 = 72 nM T02506 C7WBV5 21355678 IC50 = 53.6 nM T02506 CUL35V 21433016 IC50 = 79 nM T02506 C0HG2O 21625144 EC50 > 10000 nM T02506 C4BON1 21628493 EC50 = 0.028 nM T02506 CY56XC 21868866 EC50 = 0.3 nM T02506 C0AVF8 21868918 IC50 = 3 nM T02506 C6MTN2 21959300 IC50 = 23 nM T02506 CQS75R 22064611 Ki = 29 nM T02506 C89GZT 22221606 IC50 = 625 nM T02506 C5R3ZU 22221614 IC50 = 263 nM T02506 CD52LR 22221618 IC50 = 103 nM T02506 CU3E0Q 22221630 IC50 = 109 nM T02506 CN94JH 22221634 IC50 = 49 nM T02506 CC6X3H 22600576 IC50 > 10000 nM T02506 CT8Q2E 23349396 IC50 = 115 nM T02506 C7W5VE 23424169 IC50 = 7980 nM T02506 C6TJY8 23509070 EC50 = 16.2 nM T02506 C9O6RB 23596322 Ki > 5000 nM T02506 C8FN7B 23648275 IC50 = 17.2 nM T02506 C4TNI0 23648457 Ki = 126 nM T02506 CZGS14 23648464 Ki = 2.82 nM T02506 CBL4I8 23648465 Ki = 27.2 nM T02506 CK0XL8 23648466 Ki = 147 nM T02506 C0GP7Q 23653178 IC50 = 2650 nM T02506 CV04HC 23653179 IC50 = 1630 nM T02506 CPR38W 24015539 EC50 = 5950 nM T02506 CTE1N2 24748569 EC50 > 10000 nM T02506 C4WYE7 24749678 Ki > 1100 nM T02506 C2QHO3 24749808 Ki > 1100 nM T02506 CP7M4B 24768258 EC50 = 1000 nM T02506 CH4QT2 24768259 EC50 > 1000 nM T02506 C8DS1F 24825443 IC50 = 100 nM T02506 CZ4P8I 24825444 IC50 = 200 nM T02506 C7PR1H 24825445 IC50 = 25 nM T02506 CZ9O3D 24825446 IC50 = 1 nM T02506 CW43SX 24825447 IC50 = 13 nM T02506 CKW98C 24825448 IC50 = 10 nM T02506 CN9TA0 24825453 IC50 = 250 nM T02506 CF1H9X 24825454 IC50 = 79 nM T02506 C2PGW1 24896626 IC50 = 1440 nM T02506 C06PDG 24952192 Ki = 2300 nM T02506 CG1CF9 24952193 Ki = 5500 nM T02506 CZC7L8 24953162 IC50 > 10000 nM T02506 C4W7BN 24954947 IC50 > 10000 nM T02506 C6XC2R 24954951 IC50 > 20000 nM T02506 CHY0D7 25013322 IC50 > 10000 nM T02506 C0TPS5 25013653 IC50 > 10000 nM T02506 CWU91M 25013811 IC50 > 10000 nM T02506 CSH29L 25013812 IC50 > 10000 nM T02506 C7J6IQ 25027904 EC50 > 100000 nM T02506 C4EGR5 25027907 IC50 = 2950 nM T02506 CDK06N 25027908 IC50 = 1410 nM T02506 CKY0G2 25028122 IC50 = 32100 nM T02506 C2G1JK 25053351 Ki > 30000 nM T02506 CAW8M0 25070694 IC50 > 10000 nM T02506 CYVP87 25110671 IC50 = 8.4 nM T02506 CTYA32 25110672 IC50 = 10.4 nM T02506 CO41GX 25128805 Ki > 1000000 nM T02506 C4EI0A 25128806 Ki > 1000000 nM T02506 CQ34ZE 25128807 IC50 = 2100 nM T02506 CI19MZ 25128808 Ki > 1000000 nM T02506 COWS64 25128809 Ki > 1000000 nM T02506 C42RCW 25128810 Ki > 1000000 nM T02506 C8Q5ZK 25128811 Ki > 1000000 nM T02506 CD3Q4U 25128812 IC50 > 1000000 nM T02506 C6V1ZT 25128813 Ki > 1000000 nM T02506 CAG08U 25128815 IC50 > 1000000 nM T02506 C2FQX9 25128816 IC50 > 1000000 nM T02506 C1HLM6 25129159 Ki > 1000000 nM T02506 C7QFR2 25129160 Ki > 1000000 nM T02506 C1PS3N 25129161 Ki > 1000000 nM T02506 CZS7Q1 25129163 Ki > 1000000 nM T02506 C1XZ5O 25129164 Ki > 1000000 nM T02506 C4YMG0 25129166 Ki > 1000000 nM T02506 CX70KG 25129167 Ki = 2400 nM T02506 CGYS93 25129168 IC50 = 6900 nM T02506 C2E7NK 25129501 Ki > 1000000 nM T02506 CP7YX6 25129502 Ki > 1000000 nM T02506 CTX93Q 25129503 Ki > 1000000 nM T02506 CRA61L 25129504 Ki > 1000000 nM T02506 CV4AP7 25129505 Ki > 1000000 nM T02506 CZF6G7 25129855 Ki > 1000000 nM T02506 CNE47Z 25129856 IC50 = 1800 nM T02506 CC7FL0 25129857 IC50 = 4100 nM T02506 CV0W4X 25129858 IC50 > 1000000 nM T02506 C6W5KP 25129859 IC50 > 1000000 nM T02506 C9Z1YD 25129860 Ki > 1000000 nM T02506 CJ35NZ 25130215 Ki > 1000000 nM T02506 C2X5HD 25130216 Ki > 1000000 nM T02506 C94OVU 25130220 Ki > 1000000 nM T02506 C03ICO 25130561 Ki > 1000000 nM T02506 CZAN43 25130562 IC50 > 1000000 nM T02506 C0IFU7 25130563 IC50 > 1000000 nM T02506 CJT49R 25130564 Ki > 1000000 nM T02506 CRSM67 25130565 IC50 > 1000000 nM T02506 CM8YT4 25130566 IC50 > 1000000 nM T02506 CQ90UO 25130567 Ki > 1000000 nM T02506 COS0E1 25130893 IC50 > 1000000 nM T02506 CR29KD 25130894 IC50 > 1000000 nM T02506 CKX9J5 25130897 Ki > 1000000 nM T02506 CE9LJ6 25130898 Ki > 1000000 nM T02506 CV7WC6 25130899 Ki > 1000000 nM T02506 CJ4AK0 25130900 Ki > 1000000 nM T02506 C7HYX1 25131213 Ki > 1000000 nM T02506 C5PBM7 25131214 Ki = 7200 nM T02506 C14WCP 25131215 IC50 > 1000000 nM T02506 C7MVU3 25131217 Ki > 1000000 nM T02506 C1ZK7W 25131539 IC50 > 1000000 nM T02506 CBGD76 25131540 IC50 = 5500 nM T02506 CX3NA8 25131542 Ki > 1000000 nM T02506 CX12DM 25131544 Ki > 1000000 nM T02506 CIQ2E4 25131893 IC50 = 2100 nM T02506 C28UOB 25131894 IC50 > 1000000 nM T02506 CK2ZT3 25131895 Ki > 1000000 nM T02506 CD13ZC 25131898 IC50 > 1000000 nM T02506 C1UZL6 25132248 Ki > 1000000 nM T02506 CIO06J 25132250 IC50 = 12000 nM T02506 CVFZ60 25132251 Ki > 1000000 nM T02506 CZX45O 25132598 IC50 = 4500 nM T02506 C2ANY3 25132599 Ki > 1000000 nM T02506 CC95RT 25132600 IC50 > 1000000 nM T02506 C27KJG 25132602 IC50 > 1000000 nM T02506 CQNY78 25132933 IC50 = 6900 nM T02506 C6A8WM 25132934 IC50 > 1000000 nM T02506 CO84WJ 25132935 IC50 > 1000000 nM T02506 C6Z4IK 25132936 IC50 > 1000000 nM T02506 C9JI7L 25132937 IC50 > 1000000 nM T02506 CMYZ51 25132938 IC50 > 1000000 nM T02506 CXO4C6 25132939 Ki > 1000000 nM T02506 C9DU6Q 25132940 IC50 > 1000000 nM T02506 CZE3J7 25132941 Ki > 1000000 nM T02506 CR6ME8 25133259 Ki > 1000000 nM T02506 C0ET3J 25133260 Ki > 1000000 nM T02506 CK3VF4 25133261 Ki > 1000000 nM T02506 CB9K2T 25133267 Ki > 1000000 nM T02506 C6ZXQ0 25133268 Ki > 1000000 nM T02506 C9K0ZI 25133269 IC50 > 1000000 nM T02506 C4RG8X 25133607 Ki > 1000000 nM T02506 CD3IH0 25133608 IC50 > 1000000 nM T02506 CI82HF 25133609 IC50 = 9800 nM T02506 CM7VK8 25133611 Ki > 1000000 nM T02506 CD0NT6 25133612 Ki > 1000000 nM T02506 CWC8R0 25133614 IC50 = 5800 nM T02506 C2OCQ5 25133615 Ki = 2400 nM T02506 CEC4P2 25133616 Ki > 1000000 nM T02506 CJ98GU 25133950 Ki > 1000000 nM T02506 C32UKW 25133951 IC50 > 1000000 nM T02506 CE1WN2 25133952 Ki > 1000000 nM T02506 CNU20J 25133953 Ki > 1000000 nM T02506 C0V3KC 25133954 IC50 > 1000000 nM T02506 CLT57Z 25133955 Ki > 1000000 nM T02506 CCW71Z 25133956 Ki > 1000000 nM T02506 CA76HY 25133959 Ki > 1000000 nM T02506 CI3RZ8 25133960 IC50 > 1000000 nM T02506 C21XDY 25145083 Ki > 10000 nM T02506 CLZB04 25147765 IC50 = 37000 nM T02506 C2TJ3P 25191004 IC50 = 1000 nM T02506 C98JQI 25218466 IC50 > 10000 nM T02506 CR8F9X 25218467 IC50 > 10000 nM T02506 C87ARD 25225237 IC50 = 50000 nM T02506 CLY9W3 25235364 IC50 > 10000 nM T02506 C3FW0Y 25257459 IC50 > 10000 nM T02506 CY6X2V 25258136 IC50 = 89 nM T02506 CV4Y6N 25258138 IC50 = 93 nM T02506 CLX0P9 25258381 IC50 > 10000 nM T02506 CNLS64 25258386 IC50 = 3400 nM T02506 CSG7P9 25258611 IC50 = 670 nM T02506 COM4U3 42609838 EC50 = 170000 nM T02506 CH6PI0 43135503 IC50 = 479 nM T02506 CX89HM 44138106 Ki > 5000 nM T02506 C42TWL 44224340 EC50 = 440 nM T02506 C36BKU 44224542 EC50 = 0.11 nM T02506 C0FRP9 44224543 EC50 = 16 nM T02506 CEFT15 44224544 EC50 = 0.11 nM T02506 CLT65I 44225214 EC50 = 10.7 nM T02506 CS5PK0 44225454 EC50 = 20.2 nM T02506 CL1YK5 44225696 EC50 = 2 nM T02506 CFI64J 44227599 EC50 = 330 nM T02506 CXV83I 44227600 EC50 = 65 nM T02506 C40MCV 44275590 IC50 = 366 nM T02506 CY8L2T 44275591 IC50 = 91 nM T02506 CY1O5L 44280253 IC50 = 652 nM T02506 CHWV93 44280284 IC50 = 14 nM T02506 C3DS6O 44280299 IC50 = 490 nM T02506 CB32JI 44280300 IC50 = 89 nM T02506 CP8D0O 44280322 IC50 = 49 nM T02506 CFW6Y4 44280362 IC50 = 531 nM T02506 CTB5L8 44280369 IC50 = 109 nM T02506 C2FE9I 44280602 IC50 = 1415 nM T02506 C5PKE0 44280604 IC50 = 3563 nM T02506 CD94FC 44280669 IC50 = 1050 nM T02506 C7SY2D 44280670 IC50 = 551 nM T02506 C8YM6T 44280672 IC50 = 179 nM T02506 C6UQO3 44280673 IC50 = 68 nM T02506 CFG0A5 44280682 IC50 = 6.7 nM T02506 C9C6HY 44280687 IC50 = 929 nM T02506 C8HK7P 44280689 IC50 = 413 nM T02506 C0LNF3 44280705 IC50 = 71 nM T02506 CEX2O1 44280720 IC50 = 149 nM T02506 CKUI19 44280721 IC50 = 58 nM T02506 CPB4K1 44280724 IC50 = 105 nM T02506 C8QZY6 44283478 EC50 = 770 nM T02506 C9R3AO 44299445 Ki = 37 nM T02506 CT2MK0 44299446 Ki = 170 nM T02506 C5B6IN 44300330 IC50 = 3200 nM T02506 CH4PU5 44305819 IC50 > 10000 nM T02506 CP6A0S 44309223 IC50 = 10 nM T02506 CP52NB 44309415 IC50 = 6.2 nM T02506 CKG5Z0 44317015 IC50 > 5000 nM T02506 C2KD4V 44317238 IC50 = 1260 nM T02506 CPKH32 44317395 IC50 = 1550 nM T02506 C2GZJ0 44317407 IC50 > 5000 nM T02506 CW21CA 44317747 Ki > 10000 nM T02506 C1HK7V 44319061 Ki = 0.36 nM T02506 CE9J8B 44319062 Ki = 2.5 nM T02506 C13KXZ 44319097 Ki = 3.8 nM T02506 CX6S1W 44319117 Ki = 60 nM T02506 C28JXF 44319637 IC50 = 7 nM T02506 C7S5JR 44319707 IC50 = 7.5 nM T02506 C58TKM 44319799 IC50 = 8.8 nM T02506 C7IXG8 44319951 IC50 = 3.9 nM T02506 C8GAE7 44319960 IC50 = 3 nM T02506 C4BID0 44319971 IC50 = 2.6 nM T02506 C4XTK5 44319973 IC50 = 11 nM T02506 CC5QD0 44319981 IC50 = 3 nM T02506 CXZP05 44320014 IC50 = 35 nM T02506 CIC5N6 44320017 IC50 = 542 nM T02506 C7PS6E 44320029 IC50 = 7.4 nM T02506 CMLT05 44320030 IC50 = 490 nM T02506 CRBN05 44325311 IC50 = 5.9 nM T02506 CD0IH3 44325322 IC50 = 112 nM T02506 CNP05V 44325337 IC50 = 2 nM T02506 COTS43 44325352 IC50 = 120 nM T02506 C2B1OU 44325368 IC50 = 20.1 nM T02506 CZ9Y1O 44325433 IC50 > 3200 nM T02506 C5V7WZ 44325464 IC50 = 8 nM T02506 CS3R4P 44325467 IC50 = 53.1 nM T02506 C6NAY0 44325476 IC50 = 44.3 nM T02506 COL02R 44325510 IC50 = 341.9 nM T02506 CZ0P9W 44325539 IC50 = 34.9 nM T02506 CR94YN 44325546 IC50 = 25 nM T02506 C6TZA9 44325547 IC50 = 0.51 nM T02506 CML6J0 44325551 IC50 = 1.2 nM T02506 CL95JC 44325552 IC50 = 4.7 nM T02506 CDK3S0 44325556 IC50 = 0.5 nM T02506 CH8P0Z 44325557 IC50 = 23.1 nM T02506 C9DA8B 44325570 IC50 = 1 nM T02506 C6B7RO 44325581 IC50 = 0.8 nM T02506 C49BSH 44325582 IC50 = 14.8 nM T02506 CDX49O 44325585 IC50 = 13.5 nM T02506 CEAL30 44325586 IC50 = 5.3 nM T02506 CISM83 44325587 IC50 = 5.3 nM T02506 C8LG6M 44325589 IC50 = 1.3 nM T02506 C4K0RZ 44325613 IC50 = 1.4 nM T02506 CVD76C 44325614 IC50 = 41.1 nM T02506 CXYC85 44325632 IC50 = 3.4 nM T02506 CAE3Y9 44325639 IC50 = 0.8 nM T02506 C4S9ZI 44325650 IC50 = 1.2 nM T02506 CMJ0Z5 44325659 IC50 = 4.7 nM T02506 CEN5R9 44325692 IC50 = 1 nM T02506 CD9P3O 44343122 EC50 = 4 nM T02506 CQ7V0U 44343261 EC50 > 10000 nM T02506 C1SG7C 44348079 IC50 = 0.7 nM T02506 CSVW34 44348099 IC50 = 4.4 nM T02506 C1H7MO 44348132 IC50 = 1 nM T02506 CE4YL7 44348273 IC50 = 4 nM T02506 C28EVO 44348377 IC50 = 155 nM T02506 C2GL8B 44348457 IC50 = 21 nM T02506 CXY05L 44348479 IC50 = 3.6 nM T02506 CWCS52 44348487 IC50 = 4 nM T02506 CQA68R 44348495 IC50 = 3.6 nM T02506 CE3O6Y 44348510 IC50 = 15 nM T02506 C0I9FH 44348522 IC50 = 1.4 nM T02506 CLX35U 44348531 IC50 = 1.7 nM T02506 CX82TV 44348539 IC50 = 1 nM T02506 C90INV 44348540 IC50 = 2.3 nM T02506 C3B6LK 44355916 EC50 = 0.064 nM T02506 CK1UW9 44355917 EC50 = 5.2 nM T02506 CBO3X2 44355927 EC50 = 130 nM T02506 CIWX06 44356135 EC50 = 150 nM T02506 CW67AN 44356136 EC50 = 14 nM T02506 CM7H1I 44356536 EC50 = 73 nM T02506 C7UH6W 44356621 Ki = 13 nM T02506 CYBO90 44356823 Ki = 24 nM T02506 C4UTM7 44356833 Ki = 23 nM T02506 CT07FI 44389476 EC50 = 141 nM T02506 CG80UZ 44389487 EC50 = 21 nM T02506 CL92HF 44389493 EC50 = 59 nM T02506 COW1E9 44389558 EC50 = 19 nM T02506 C5ECY2 44389569 EC50 = 92 nM T02506 CY5K2O 44389570 EC50 = 173 nM T02506 CRN5I1 44389572 EC50 = 143 nM T02506 CL7C9P 44389577 EC50 = 2411 nM T02506 CZJ5C4 44389581 EC50 = 1.6 nM T02506 C9Q4UB 44389582 EC50 = 1 nM T02506 CSP4T9 44389593 EC50 = 137 nM T02506 CEHT06 44389595 EC50 = 0.6 nM T02506 CTJ9Q6 44389606 EC50 = 743 nM T02506 CS47PF 44389609 EC50 = 2.6 nM T02506 CUA5F4 44389617 EC50 = 36 nM T02506 CVT09Q 44389633 EC50 = 336 nM T02506 CV24GJ 44389648 EC50 = 1980 nM T02506 C8MI1L 44389650 EC50 = 203 nM T02506 C9RUX6 44389654 EC50 = 43 nM T02506 CL2W9P 44389655 EC50 = 68 nM T02506 CQ01VW 44389659 EC50 = 50 nM T02506 C2PDC8 44389876 IC50 = 0.86 nM T02506 C8ZIP3 44389878 IC50 = 1.72 nM T02506 CA05VL 44389880 IC50 = 2.12 nM T02506 CB1H3E 44389883 IC50 = 1.39 nM T02506 CUP57N 44389890 IC50 = 14.46 nM T02506 CBIA52 44389891 IC50 = 2.15 nM T02506 CQU8C6 44389896 IC50 = 2.65 nM T02506 C10LSB 44389901 IC50 = 3.05 nM T02506 C6CIB9 44389904 IC50 = 1.43 nM T02506 C8YNX2 44389906 IC50 = 0.22 nM T02506 C39DPH 44389907 IC50 = 3.58 nM T02506 C2ZS9G 44389914 IC50 = 2.74 nM T02506 C19MKQ 44389919 IC50 = 3.94 nM T02506 C4W5VU 44389922 IC50 = 0.43 nM T02506 CB7K5Y 44389934 IC50 = 0.46 nM T02506 CVG41F 44389943 IC50 = 0.27 nM T02506 CO1H5G 44389945 IC50 = 1.08 nM T02506 C8GD3V 44389948 IC50 = 0.22 nM T02506 CP0Y8G 44390069 IC50 = 1.4 nM T02506 C1JQD2 44390070 IC50 = 38 nM T02506 CPFB84 44390071 IC50 = 0.3 nM T02506 C24ZDP 44390072 IC50 = 0.9 nM T02506 CXHL23 44390084 IC50 = 14 nM T02506 CQ92BW 44390097 IC50 = 0.9 nM T02506 C6RC2Y 44390116 IC50 = 45 nM T02506 C4GP0U 44390120 IC50 = 0.8 nM T02506 C1DS5R 44390163 IC50 = 0.8 nM T02506 C7ZQ1J 44391057 IC50 = 39 nM T02506 C50XAP 44391076 IC50 = 13 nM T02506 C5Y6CT 44391206 IC50 = 2.4 nM T02506 C0ZIT7 44391782 IC50 = 0.3 nM T02506 CS4XD9 44391788 IC50 = 6.3 nM T02506 CV4G0H 44391842 IC50 = 0.7 nM T02506 CRJE53 44391854 IC50 = 0.4 nM T02506 C5W2IH 44391860 IC50 = 2.5 nM T02506 CZOJ29 44391870 IC50 = 0.5 nM T02506 CIT5P8 44391879 IC50 = 1.7 nM T02506 C0B5IT 44391881 IC50 = 0.7 nM T02506 CZH85I 44391888 IC50 = 1.2 nM T02506 CQD42M 44391889 IC50 = 0.9 nM T02506 CT0BO6 44391890 IC50 = 0.8 nM T02506 C1NIS3 44391905 IC50 = 0.7 nM T02506 C74EHI 44391917 IC50 = 0.5 nM T02506 CP15SF 44392410 IC50 = 19.82 nM T02506 CA82NU 44392580 IC50 = 990 nM T02506 CC72ZY 44392593 IC50 = 335 nM T02506 CDMN93 44392636 IC50 = 12 nM T02506 CS8ZN5 44393200 IC50 = 1.2 nM T02506 CP53NK 44393219 IC50 = 0.8 nM T02506 CB5DS4 44393237 IC50 = 1 nM T02506 C1GA9N 44393240 IC50 = 1.7 nM T02506 C0TLH5 44393249 IC50 = 2.2 nM T02506 CL27NW 44393263 IC50 = 0.3 nM T02506 CR64AD 44393267 IC50 = 0.5 nM T02506 CTN81R 44393286 IC50 = 0.9 nM T02506 CW59RL 44393287 IC50 = 2.5 nM T02506 C01ODV 44393310 IC50 = 0.6 nM T02506 C82WUF 44393322 IC50 = 2 nM T02506 CO1Q0W 44393335 IC50 = 0.6 nM T02506 C0JXU4 44393336 IC50 = 1.5 nM T02506 CC89WN 44393340 IC50 = 0.4 nM T02506 C2WXI0 44393342 IC50 = 3.9 nM T02506 CNP73S 44393366 IC50 = 0.6 nM T02506 C8E0AJ 44393367 IC50 = 2.2 nM T02506 CQY82B 44393380 IC50 = 0.6 nM T02506 CP25CW 44393381 IC50 = 1.8 nM T02506 C8P3FU 44393399 IC50 = 1.3 nM T02506 CIS79C 44393400 IC50 = 2 nM T02506 C1XOK4 44393405 IC50 = 0.5 nM T02506 CV5YB6 44393408 IC50 = 7.3 nM T02506 CRB41V 44393419 IC50 = 16 nM T02506 C5U2KP 44394160 IC50 = 209 nM T02506 C13SYV 44396250 Ki = 19 nM T02506 CB1P0S 44396251 Ki = 8.8 nM T02506 CHY1C3 44396271 Ki = 72 nM T02506 C29MBI 44396272 Ki = 11 nM T02506 C4TQ6N 44396282 Ki = 11 nM T02506 CH2Y3L 44396283 Ki = 6.2 nM T02506 CWZB52 44396284 Ki = 140 nM T02506 CD80LM 44396296 Ki = 34 nM T02506 C6SI5L 44396297 Ki > 200 nM T02506 C45LRH 44396317 Ki = 10 nM T02506 C5JG6H 44396330 Ki = 46 nM T02506 CA8V4G 44396331 Ki = 94 nM T02506 CD2EY3 44399091 IC50 > 5000 nM T02506 CDJ7H0 44399199 IC50 = 1800 nM T02506 CK1X0O 44400690 IC50 = 877 nM T02506 CSE07P 44402388 IC50 = 3.34 nM T02506 CSZ2J0 44402418 IC50 = 31.2 nM T02506 C6I3PD 44402432 IC50 = 27.2 nM T02506 C3FR5B 44402483 IC50 = 18 nM T02506 C6CWQ3 44402516 IC50 = 10 nM T02506 CC3QK6 44402532 IC50 = 57.4 nM T02506 CM35QL 44402545 IC50 = 18 nM T02506 CL9CQ8 44402598 IC50 = 51.4 nM T02506 CN57AQ 44402634 IC50 = 126 nM T02506 CQH5B1 44402654 IC50 = 6 nM T02506 CF0VN8 44402705 IC50 = 39 nM T02506 C7VCZ5 44402711 IC50 > 10000 nM T02506 CXI97U 44402746 IC50 > 10000 nM T02506 CGRX27 44402769 IC50 > 10000 nM T02506 C9XS4E 44402799 IC50 > 10000 nM T02506 CB2V0A 44403942 Ki = 7.3 nM T02506 CARV69 44405133 IC50 = 0.6 nM T02506 CKZ15D 44405150 IC50 = 0.5 nM T02506 CR4V3M 44405163 IC50 = 0.6 nM T02506 C2C9OW 44405166 IC50 = 0.2 nM T02506 CG85OU 44405167 IC50 = 0.5 nM T02506 CLE8X1 44405174 IC50 = 0.4 nM T02506 C72SFE 44405903 IC50 = 1730 nM T02506 CB56DO 44407581 IC50 = 830 nM T02506 CWT4M0 44407582 EC50 = 830 nM T02506 C1ISP9 44407583 EC50 = 153 nM T02506 C5WQ6O 44407584 IC50 = 16 nM T02506 CP5DT4 44407585 IC50 = 14 nM T02506 C2A5EY 44407586 EC50 = 12 nM T02506 C79JEI 44407631 EC50 = 160 nM T02506 CB0L6S 44407636 EC50 = 1000 nM T02506 C2W0PF 44407655 EC50 > 1000 nM T02506 CA7S2Z 44407657 EC50 = 378 nM T02506 CWU1O4 44407658 IC50 = 5155 nM T02506 CP7CQ0 44407661 EC50 = 480 nM T02506 CNC2A4 44407662 IC50 = 26 nM T02506 CCPB47 44407663 IC50 = 60 nM T02506 C8Y7ZB 44407724 IC50 = 328 nM T02506 C5QW0O 44407725 EC50 = 1391 nM T02506 C3LGU8 44407741 IC50 = 892 nM T02506 C6J3VA 44407760 EC50 = 3237 nM T02506 C1O6WJ 44407763 EC50 = 583 nM T02506 C21CBM 44407771 EC50 = 844 nM T02506 CD3E0R 44407782 EC50 > 1000 nM T02506 C2O1DA 44407785 IC50 = 3984 nM T02506 C2POZ8 44407805 IC50 = 109 nM T02506 CQ1Y0R 44407807 EC50 = 161 nM T02506 CZ0XT5 44407808 EC50 = 144 nM T02506 CF5Z0G 44407811 EC50 = 650 nM T02506 CF0AQ2 44407812 EC50 = 243 nM T02506 CN06HP 44407826 IC50 = 253 nM T02506 CUA05F 44407827 EC50 = 63 nM T02506 CXD31Y 44407857 EC50 > 1000 nM T02506 C4K3ZG 44408764 IC50 = 157 nM T02506 C7CSE3 44408771 IC50 = 5460 nM T02506 CF06GJ 44408808 IC50 = 524 nM T02506 C1K3FC 44409005 IC50 = 229 nM T02506 C5HM2W 44409078 IC50 = 1090 nM T02506 CIUR71 44409233 IC50 > 10000 nM T02506 CF0IQ7 44412807 IC50 > 10000 nM T02506 CI4KN9 44412821 IC50 = 1420 nM T02506 C5E9XO 44412823 IC50 = 880 nM T02506 C5S9OV 44412835 IC50 = 3740 nM T02506 CN9X6E 44412848 IC50 > 10000 nM T02506 CE60QX 44412849 IC50 = 481 nM T02506 CZ13IC 44412903 IC50 = 113 nM T02506 C3ADY8 44412904 IC50 = 389 nM T02506 CJ4S8E 44412954 IC50 = 4245 nM T02506 C0JAX2 44412955 IC50 > 10000 nM T02506 C4EZB6 44412956 IC50 = 319 nM T02506 CW08IO 44412979 IC50 = 6450 nM T02506 CFH31O 44412983 IC50 = 79 nM T02506 C5RT0I 44413033 IC50 = 567 nM T02506 C2TFX6 44413049 IC50 > 10000 nM T02506 CE2P7W 44413050 IC50 = 4023 nM T02506 CQW1N9 44414035 IC50 = 46 nM T02506 CXBZ80 44414036 EC50 = 33.1 nM T02506 C2H8RD 44414046 IC50 = 93 nM T02506 CQC9F4 44414050 EC50 = 1170 nM T02506 CIS2L0 44414060 EC50 = 152 nM T02506 CJBQ27 44414066 EC50 = 61 nM T02506 C09CRE 44414068 IC50 = 1478 nM T02506 CECT78 44414069 IC50 = 2080 nM T02506 CI12OU 44414094 EC50 = 50 nM T02506 CF5T6Y 44414110 IC50 = 176 nM T02506 CGP27O 44414111 IC50 = 470 nM T02506 CXG13L 44414126 EC50 = 104 nM T02506 C8E5PN 44414131 EC50 = 65 nM T02506 CV1LR4 44414182 IC50 = 230 nM T02506 CALJ60 44414245 IC50 = 23 nM T02506 C5WTR2 44414246 IC50 = 49.2 nM T02506 C7MT9J 44414260 IC50 = 139 nM T02506 CL0K4C 44414274 IC50 = 40 nM T02506 C90LXU 44414284 EC50 = 1100 nM T02506 C0I3YZ 44414292 IC50 = 422 nM T02506 CPFS03 44414293 IC50 = 82 nM T02506 C7L2PW 44415352 IC50 = 1210 nM T02506 C2Y9BF 44415353 IC50 = 455 nM T02506 C96JSR 44415397 IC50 = 3900 nM T02506 C5V2SP 44415478 IC50 = 97 nM T02506 C7YQ9X 44415498 IC50 = 414 nM T02506 CREK89 44415499 IC50 = 146 nM T02506 C18JCA 44415511 IC50 = 310 nM T02506 CGS79I 44415523 IC50 = 84 nM T02506 C1FCL0 44415547 IC50 = 605 nM T02506 C6PD3R 44415553 EC50 = 169 nM T02506 CH50DC 44415571 EC50 = 79 nM T02506 CSF5O8 44415669 EC50 = 241 nM T02506 C7C4XF 44415699 EC50 = 391 nM T02506 CCO34X 44415700 EC50 = 30 nM T02506 C3KI0H 44415761 IC50 > 10000 nM T02506 CV37CW 44415788 EC50 = 140 nM T02506 C9T3QO 44423844 EC50 = 100 nM T02506 CG72WC 44427370 Ki = 0.4 nM T02506 C2F8CW 44427371 Ki = 0.73 nM T02506 CHB94D 44427372 Ki = 0.24 nM T02506 CYB7J6 44427373 Ki = 0.18 nM T02506 CQ96LY 44427374 Ki = 0.2 nM T02506 CN2M3P 44427375 Ki = 1.09 nM T02506 CQ74SE 44427404 Ki = 0.091 nM T02506 CHK6A4 44427405 Ki = 0.48 nM T02506 CL1Y4N 44430357 IC50 = 3300 nM T02506 C5S6XP 44430360 IC50 = 2470 nM T02506 CUQT28 44430361 IC50 > 5000 nM T02506 CKF6I1 44430362 IC50 > 5000 nM T02506 COT67E 44430364 IC50 = 802 nM T02506 C2YF4G 44430366 IC50 = 2640 nM T02506 CBGX08 44430369 IC50 > 5000 nM T02506 CY4XR5 44430372 IC50 = 21 nM T02506 C27KUN 44430374 IC50 = 802 nM T02506 C6LV9A 44430376 IC50 = 53 nM T02506 CHM5G2 44430378 IC50 > 5000 nM T02506 C4ERT8 44433138 Ki = 7100 nM T02506 C9EK6V 44433139 Ki = 12000 nM T02506 CEJ8B1 44433140 Ki = 32000 nM T02506 CNX1A6 44433141 Ki = 7900 nM T02506 C2J1PU 44433142 Ki = 38000 nM T02506 C3SJ5V 44433504 Ki > 1100 nM T02506 CJ5G2Z 44439806 IC50 = 11 nM T02506 CG17VZ 44439807 IC50 = 1 nM T02506 C5Y4CM 44439809 IC50 = 37 nM T02506 C28PCX 44439811 IC50 = 1134 nM T02506 C4WS3E 44439813 IC50 = 378 nM T02506 C3H6BA 44439815 IC50 = 40 nM T02506 C3DGB7 44439820 IC50 = 31 nM T02506 CL9IE2 44439822 IC50 = 6.6 nM T02506 C7RLX5 44439823 IC50 = 13 nM T02506 C1A0PH 44439825 IC50 = 10.1 nM T02506 C3KS9O 44439826 IC50 = 22 nM T02506 CFZ0N1 44439827 IC50 = 9.1 nM T02506 CMW5Z8 44439828 IC50 = 440 nM T02506 CWBD12 44439829 IC50 = 69 nM T02506 C2Y4GR 44439830 IC50 = 23 nM T02506 CZNS72 44439831 IC50 = 13 nM T02506 COGW71 44439832 IC50 = 20 nM T02506 C76TMP 44439833 IC50 = 175 nM T02506 C82NQD 44439834 IC50 = 7.8 nM T02506 C98BPO 44439835 IC50 = 4.9 nM T02506 C1HZ2K 44439836 IC50 = 4 nM T02506 C3LO1U 44440237 EC50 = 980 nM T02506 CLK05T 44440238 IC50 = 2330 nM T02506 CP3JU8 44440239 EC50 > 1000 nM T02506 C34ERB 44440240 EC50 = 4893 nM T02506 C5KG7L 44440241 EC50 = 1300 nM T02506 CB1ZS3 44440262 EC50 = 44 nM T02506 CKON02 44440263 EC50 = 435 nM T02506 C5DB8N 44440264 EC50 > 1000 nM T02506 C89JEW 44440265 EC50 > 1000 nM T02506 CR7G2K 44440266 EC50 > 1000 nM T02506 CVT4O9 44440267 EC50 > 1000 nM T02506 CO98DZ 44440268 EC50 > 1000 nM T02506 CC73BF 44440269 EC50 = 407 nM T02506 C6O5DS 44441690 Ki = 37 nM T02506 C8YOH7 44441691 Ki = 100 nM T02506 CG6W1K 44441692 Ki = 35 nM T02506 C5OMR2 44441693 Ki = 75 nM T02506 CKQ1H7 44441694 Ki = 332 nM T02506 CEMX26 44441695 Ki = 63052 nM T02506 C5WVG8 44441696 Ki = 382 nM T02506 CY32PU 44441697 Ki = 17879 nM T02506 CL3WI5 44441857 IC50 = 5300 nM T02506 CIL2C9 44441858 EC50 > 1000 nM T02506 CR2S3A 44441859 IC50 = 3110 nM T02506 C6GRK9 44441860 EC50 > 1000 nM T02506 C2FC5N 44441861 EC50 = 820 nM T02506 CA1BY2 44441862 IC50 = 4380 nM T02506 C6SMB2 44441863 EC50 = 490 nM T02506 CTQ15A 44441864 EC50 > 1000 nM T02506 CF06VH 44441865 EC50 = 130 nM T02506 C1X5MS 44441866 EC50 = 430 nM T02506 CYG7X4 44473146 IC50 > 10000 nM T02506 CT0B2Q 44473422 EC50 > 1000 nM T02506 CR5SI0 44476535 EC50 > 10000 nM T02506 CM29JD 44516036 IC50 > 10000 nM T02506 C3ND5A 44542643 EC50 > 1000 nM T02506 C3SBL5 44543099 EC50 > 1000 nM T02506 CK8MH3 44565647 Ki = 26300 nM T02506 CEI26D 44569027 Ki > 1000000 nM T02506 CCPW27 44569028 IC50 > 1000000 nM T02506 CF4RS6 44569029 Ki = 7500 nM T02506 CEA0U9 44579680 Ki = 55 nM T02506 C8W6ZF 44580025 Ki = 977 nM T02506 CXGP15 44580026 Ki = 724 nM T02506 CW5O3K 44580027 Ki = 158 nM T02506 C2L3NV 44588414 IC50 = 16000 nM T02506 C3TRJ2 44589610 EC50 = 10 nM T02506 CZOU20 44589952 IC50 = 8.77 nM T02506 CNM79D 44589953 IC50 = 1.9 nM T02506 C1JCM3 44589998 IC50 = 6.7 nM T02506 CDP6W8 44589999 IC50 = 10.3 nM T02506 C5FC9V 44590000 IC50 = 16.2 nM T02506 CYI29S 44590098 IC50 = 14 nM T02506 CD8R7Y 44590099 IC50 = 126 nM T02506 C7T8KP 44590100 IC50 > 15000 nM T02506 C4RZX5 44590136 IC50 = 6.5 nM T02506 C6NZW2 44590137 IC50 = 5.57 nM T02506 CL7IT6 44592556 IC50 > 100000 nM T02506 CJ3VI8 44593465 Ki > 5000 nM T02506 C6NXD9 44593529 IC50 = 5500 nM T02506 CKYW84 44596355 IC50 = 1200 nM T02506 CY0U6X 44596356 IC50 = 150 nM T02506 CQG0F7 44596357 IC50 > 1000 nM T02506 CSR28W 44596358 IC50 > 1000 nM T02506 CAG36H 44596359 IC50 = 16 nM T02506 C6AZU3 44596467 IC50 = 5 nM T02506 C49XRU 44596468 IC50 = 293 nM T02506 C1YRA4 44596469 IC50 = 1210 nM T02506 CS12MF 44596470 IC50 = 1570 nM T02506 C2K1DR 44596471 IC50 = 3.3 nM T02506 C3LMA0 44596573 IC50 = 180 nM T02506 C3KH5Y 44596574 IC50 = 85 nM T02506 CJM37H 44596575 IC50 = 100 nM T02506 C8GJ9B 44596686 IC50 = 3.4 nM T02506 CSQ10X 44596687 IC50 = 190 nM T02506 CFJE97 44596688 IC50 = 13 nM T02506 CYX0C2 44596789 IC50 = 11.1 nM T02506 CM67OY 44596790 IC50 = 4.2 nM T02506 CUT7N3 44596791 IC50 = 6.3 nM T02506 CAI8D6 44596792 IC50 > 10000 nM T02506 C9KW4Y 44596793 IC50 = 687 nM T02506 CBLN03 44596894 IC50 > 1000 nM T02506 CX76YZ 44596895 IC50 = 9 nM T02506 CLWY41 44596896 IC50 = 4 nM T02506 CSUT20 44596897 IC50 = 35 nM T02506 CRUO49 44596898 IC50 > 1000 nM T02506 C1FI6O 44596992 IC50 = 4.5 nM T02506 C0YUC1 44596993 IC50 = 6.3 nM T02506 CN1M3J 44596994 IC50 = 128 nM T02506 C6NEV4 44596995 IC50 = 150 nM T02506 C42NEY 44596996 IC50 = 2.5 nM T02506 CUK16W 44597094 IC50 = 122 nM T02506 C43LCQ 44597095 IC50 = 10 nM T02506 CLJM84 44597096 IC50 = 161 nM T02506 C9R2CP 44597097 IC50 = 111 nM T02506 CL01OK 44597098 IC50 = 312 nM T02506 CMR68J 44597209 IC50 = 6.2 nM T02506 CWG9Z7 44597210 IC50 = 40.97 nM T02506 CYA0B6 44597211 IC50 = 580 nM T02506 CE31LY 44597212 IC50 = 590 nM T02506 C9QO1F 44597743 IC50 = 293 nM T02506 C63LWP 44597744 IC50 = 5.4 nM T02506 C3O2NE 44597745 IC50 = 217 nM T02506 CME14J 44597857 IC50 = 1.2 nM T02506 CI9E7J 44597858 IC50 = 1.6 nM T02506 C95YGF 44597859 IC50 = 1.2 nM T02506 CD9EL6 44597860 IC50 = 8.7 nM T02506 C6GWQ8 44597861 IC50 = 4.8 nM T02506 CS79YT 44597968 IC50 = 2.63 nM T02506 CUO92A 44597969 IC50 = 310 nM T02506 CMXI54 44597970 IC50 = 326 nM T02506 CT9Q0J 44597971 IC50 = 4.8 nM T02506 CSOD50 44597973 IC50 = 120 nM T02506 CIJP09 44605898 EC50 > 10000 nM T02506 C9PLK4 45263610 IC50 > 2000 nM T02506 C78JKD 45265930 IC50 > 2000 nM T02506 CN4IE3 45275362 IC50 = 8.1 nM T02506 C4A2MR 46190224 IC50 = 24400 nM T02506 CKX73S 46190225 IC50 = 7600 nM T02506 CJ3Z5R 46231169 EC50 = 27 nM T02506 C9CL7N 46231170 EC50 = 300 nM T02506 C3O2GA 46231223 EC50 = 4000 nM T02506 CR6XM0 46231224 EC50 = 2 nM T02506 C51IGU 46231225 EC50 = 4000 nM T02506 C0ZBS6 46231226 EC50 = 27 nM T02506 C4M9KI 46231227 EC50 = 1500 nM T02506 CJ84WL 46231228 EC50 = 2600 nM T02506 C5C8ZD 46237712 EC50 = 14.06 nM T02506 CP1VU0 46237713 IC50 = 243.22 nM T02506 C0HMU5 46237838 EC50 = 16.48 nM T02506 C6RZX9 46237839 EC50 = 6.918 nM T02506 CKBD82 46237840 EC50 = 92.04 nM T02506 CPD64X 46237841 EC50 = 35.97 nM T02506 C2S6PL 46834818 IC50 > 10000 nM T02506 CL6SY4 46866497 IC50 > 30000 nM T02506 CO1T3Q 46871902 IC50 = 57200 nM T02506 C9UZ5N 46871916 IC50 = 151100 nM T02506 CAYW93 46880832 Ki = 29000 nM T02506 CDHA57 46880834 IC50 > 30000 nM T02506 C72MUY 46889765 IC50 > 5000 nM T02506 C6DVO1 46889848 IC50 > 10000 nM T02506 CZ90FC 46894119 IC50 > 25000 nM T02506 C3Q7RI 46913890 IC50 > 4960 nM T02506 CX70GY 46915355 IC50 > 10000 nM T02506 CN9L7G 46916268 IC50 = 2200 nM T02506 C0FNE4 46916592 IC50 = 3.7 nM T02506 CYVP45 46916643 IC50 = 3.8 nM T02506 C05YMH 46935020 IC50 = 82 nM T02506 CL7P3N 46938234 IC50 > 10000 nM T02506 CX0NO8 49782554 EC50 < 15848.93 nM T02506 CC7T8Q 49782555 EC50 = 1655.77 nM T02506 CD07EV 49782777 EC50 < 15848.93 nM T02506 C43UKW 49782778 IC50 < 15848.93 nM T02506 C2JTF0 49782779 EC50 = 1028.02 nM T02506 CS7KX9 49782780 IC50 < 15848.93 nM T02506 C36RYU 49782781 EC50 = 402.72 nM T02506 C8OA0C 49782985 IC50 < 15848.93 nM T02506 C5Y6QU 49782986 EC50 = 35.48 nM T02506 CB8V7R 49782987 EC50 = 9954.05 nM T02506 CU3S6H 49836028 Ki > 50000 nM T02506 C96SLW 49851364 Ki > 100000 nM T02506 CDN4K6 49851369 Ki > 50000 nM T02506 C4YXN1 49851467 Ki > 50000 nM T02506 CUD91T 49862248 EC50 = 1043000 nM T02506 C0SY6G 49864608 EC50 = 0.24 nM T02506 C2JAP4 50919273 EC50 = 20000 nM T02506 C0BPT6 50919274 EC50 = 1870 nM T02506 CY10IC 50940834 EC50 > 10000 nM T02506 CTH45Q 52918523 IC50 > 10000 nM T02506 CF16DR 52937206 EC50 = 340000 nM T02506 CG7LY6 52937207 EC50 = 2300 nM T02506 CS0UY6 52937307 EC50 = 6200 nM T02506 CB94DP 52937308 EC50 = 700000 nM T02506 C75SPY 52937309 EC50 = 600000 nM T02506 CFNK21 52946352 IC50 = 310 nM T02506 CF4W1S 53262779 IC50 = 1000000 nM T02506 CA3SG5 53262780 IC50 = 80000 nM T02506 C83ZHQ 53262781 IC50 = 2800000 nM T02506 C8MU3A 53322265 IC50 > 10000 nM T02506 CYA61L 53323081 EC50 = 7 nM T02506 CEW0A8 53324900 IC50 = 8360 nM T02506 CJCP75 53359074 Ki > 75000 nM T02506 CZQ09C 53465819 IC50 = 1100 nM T02506 CWHK62 53483961 EC50 > 5400 nM T02506 C87KXG 54584962 IC50 = 3500000 nM T02506 C30XLO 54592009 IC50 > 10000 nM T02506 C5ZX4B 54597874 IC50 > 10000 nM T02506 C6ST8W 54675748 IC50 = 0.2 nM T02506 CDI89A 54765689 IC50 = 0.2 nM T02506 CB8U5G 54765691 IC50 = 0.3 nM T02506 CX0Q9I 54765856 IC50 = 0.2 nM T02506 C8O3BH 54765858 IC50 = 0.2 nM T02506 CPM43H 54765860 IC50 = 0.2 nM T02506 C4XG5H 54766021 IC50 = 0.2 nM T02506 CRLE21 54766022 IC50 = 0.2 nM T02506 C7CBA8 54766023 IC50 = 0.2 nM T02506 CJ2K9E 54766174 IC50 = 0.2 nM T02506 C3CNJ8 54766175 IC50 = 0.4 nM T02506 CLP3H4 54766176 IC50 = 0.3 nM T02506 CY5QJ4 54766177 IC50 = 0.1 nM T02506 CR5T9O 54766178 IC50 = 9.7 nM T02506 C90PVJ 54766328 IC50 = 0.4 nM T02506 CL38TD 54766331 IC50 = 0.4 nM T02506 CPH2W0 54766478 IC50 = 0.4 nM T02506 CRP5Z2 54766481 IC50 = 0.4 nM T02506 CHG78U 54766482 IC50 = 0.2 nM T02506 C8AUT4 54766633 IC50 = 0.3 nM T02506 CT7D3W 54766636 IC50 = 0.9 nM T02506 CMO2X4 54766789 IC50 = 0.5 nM T02506 CNUM98 54766945 IC50 = 0.1 nM T02506 C8GR2U 54767099 IC50 = 0.3 nM T02506 C3X1IA 54767260 IC50 = 5.7 nM T02506 C9W5DZ 56593984 Ki > 75000 nM T02506 C8GP2M 56658858 EC50 > 2680 nM T02506 C0HMP7 56662184 EC50 = 357 nM T02506 CH65JX 56662340 EC50 = 2310 nM T02506 C1WS4G 56662341 EC50 > 6510 nM T02506 CWY30K 56665645 EC50 = 3500 nM T02506 C1O0XA 56666151 IC50 = 1.11 nM T02506 CFQ51I 56672695 EC50 = 3800 nM T02506 C9CXS4 56675930 EC50 > 3200 nM T02506 CZT8H6 56676055 EC50 > 1100 nM T02506 C9ZJ8I 56679386 EC50 > 4560 nM T02506 CP06XK 56679387 EC50 > 10000 nM T02506 CP58AC 56679388 EC50 > 10000 nM T02506 CK1N6F 56682681 EC50 > 2610 nM T02506 CG8J9I 56682682 EC50 > 4800 nM T02506 C67XZQ 56927060 EC50 = 2.6 nM T02506 C51ZSU 56940798 EC50 = 0.7 nM T02506 CGK89W 56940799 EC50 = 2 nM T02506 CURV45 56940800 EC50 = 14 nM T02506 C3F0IO 56940801 EC50 = 0.8 nM T02506 C80ZVD 56940946 EC50 = 4 nM T02506 CR4TO6 56941387 EC50 = 3 nM T02506 CZ3DB1 56941388 EC50 = 49 nM T02506 C48FPW 56941825 EC50 = 4 nM T02506 CUQ8X4 56941959 EC50 = 11 nM T02506 CZD36T 56941964 EC50 = 15 nM T02506 C5UK3N 56942100 EC50 = 6 nM T02506 CUB7H1 56942101 EC50 = 28 nM T02506 CGY2K5 56942102 EC50 = 36 nM T02506 COA86V 56942249 EC50 = 3 nM T02506 CBX8N7 56942543 EC50 = 957 nM T02506 CK1G7N 56943018 EC50 = 10 nM T02506 C53OZE 56945585 EC50 = 6.2 nM T02506 C37IJX 57392620 Ki = 1 nM T02506 CF83VM 57401459 Ki > 75000 nM T02506 CTM6K5 57690900 IC50 > 5000 nM T02506 C87TXE 57992044 EC50 > 10000 nM T02506 CI6XF5 58742295 IC50 > 3200 nM T02506 CYI71B 58902727 EC50 > 10000 nM T02506 CE18JH 60202715 EC50 = 27 nM T02506 CE0SK2 66574394 IC50 < 100000 nM T02506 C26BLT 66792935 EC50 = 0.9 nM T02506 CK7C3F 66793234 EC50 = 1 nM T02506 C7D5KR 66793358 EC50 = 27 nM T02506 CW5I4N 66800025 EC50 = 200 nM T02506 CS2XF1 66800044 EC50 = 5.9 nM T02506 CC4D3G 66800191 EC50 = 22 nM T02506 CU3CO9 66800285 EC50 = 357 nM T02506 C8FG7K 66800295 EC50 = 23 nM T02506 CXA2F8 66800317 EC50 = 57 nM T02506 CVH2W8 66800328 EC50 = 6 nM T02506 C2LN5Q 66800382 EC50 = 240 nM T02506 CV63IY 66800384 EC50 = 460 nM T02506 CZLD42 66800405 EC50 = 150 nM T02506 CIGK37 66800456 EC50 = 0.7 nM T02506 CANS48 66801915 EC50 = 350 nM T02506 CRE4B8 66802205 EC50 = 6280 nM T02506 C3Z7JY 66802304 EC50 = 260 nM T02506 C3SKM2 66802363 EC50 = 110 nM T02506 CPU8J0 66802555 EC50 = 1130 nM T02506 C8C4HE 66802616 EC50 = 110 nM T02506 CZ69XC 66802706 EC50 = 101 nM T02506 C6ZF2N 66802727 EC50 = 340 nM T02506 CN07XA 66802737 EC50 > 500 nM T02506 CF3G2U 66802742 EC50 = 1.5 nM T02506 CI1G8L 66802787 EC50 > 500 nM T02506 CZ8KP0 66802802 EC50 = 160 nM T02506 CF1WN2 66803137 EC50 = 2 nM T02506 C24JEX 66803231 EC50 = 8 nM T02506 CBO20T 66803277 EC50 = 0.5 nM T02506 C2F5TS 68037237 EC50 = 17 nM T02506 CMT2I3 68321354 IC50 = 280 nM T02506 CH5F3L 68324545 IC50 = 8210 nM T02506 C7KM0T 68779769 IC50 = 3.1 nM T02506 CHVW02 69281197 EC50 = 75 nM T02506 C6XQM8 70140794 IC50 = 20 nM T02506 C5AY3Z 70261892 IC50 = 5490 nM T02506 CBM80I 70354859 EC50 = 26.9 nM T02506 C4NMI7 70681450 IC50 = 0.6 nM T02506 CID9L6 70681451 IC50 = 0.2 nM T02506 C6YL4K 70681621 EC50 = 2.8 nM T02506 CT85IV 70681622 EC50 = 110 nM T02506 CFD6Y8 70681623 EC50 = 1300 nM T02506 CMI8Q9 70681848 IC50 < 100000 nM T02506 CARO49 70685018 Ki = 14 nM T02506 CZC61P 70685893 EC50 = 2.2 nM T02506 C6G1AZ 70685894 EC50 = 14 nM T02506 CF4D0J 70685895 EC50 = 200 nM T02506 CI3RN7 70685896 EC50 = 12 nM T02506 CJ5Z4N 70686080 IC50 < 100000 nM T02506 CR0MB3 70688747 EC50 = 120 nM T02506 CLO8E7 70690044 EC50 = 110 nM T02506 CNOJ60 70690045 EC50 = 2000 nM T02506 COU7T5 70690046 EC50 = 1200 nM T02506 C1KFL5 70690047 EC50 = 3150 nM T02506 CGU65P 70690163 Ki = 2.4 nM T02506 CWGC38 70692196 EC50 = 0.14 nM T02506 CH92NS 70694259 EC50 = 1100 nM T02506 CLVB71 70694260 EC50 = 210 nM T02506 CTK9H2 70694261 EC50 = 27 nM T02506 CGOH19 70694262 EC50 = 770 nM T02506 CY7EL2 70694264 EC50 = 2250 nM T02506 CIRY65 70694390 Ki = 5.3 nM T02506 CSWT16 70696334 EC50 = 670 nM T02506 CP5QM9 70696352 EC50 = 9.2 nM T02506 CZ72LR 70696353 EC50 = 11000 nM T02506 C3PM4W 70696354 EC50 = 5500 nM T02506 CRKF46 71153846 IC50 = 32500 nM T02506 CUH71V 71239417 IC50 > 1000 nM T02506 CG24SA 71449116 IC50 = 0.97 nM T02506 CW0N5Y 71450112 EC50 = 16 nM T02506 CJ3R1C 71450113 EC50 = 0.84 nM T02506 CGWH69 71453711 EC50 = 60 nM T02506 CDV74Z 71453712 EC50 = 0.12 nM T02506 CVB70T 71453742 EC50 = 0.31 nM T02506 C59KRH 71453743 EC50 = 100 nM T02506 COPG39 71454424 EC50 = 400 nM T02506 CG5H6B 71454465 IC50 = 6000 nM T02506 C15HIA 71455440 EC50 = 1.6 nM T02506 CN76BF 71457218 EC50 = 0.4 nM T02506 C2J7BX 71457266 EC50 = 0.67 nM T02506 CUAD52 71457267 EC50 = 47 nM T02506 C8DOM0 71457268 EC50 = 15 nM T02506 C2TN5I 71458013 IC50 = 235 nM T02506 C71HUY 71459076 EC50 = 0.27 nM T02506 CR14YQ 71459915 IC50 = 1700 nM T02506 CUAG08 71460882 EC50 = 0.2 nM T02506 CN87JE 71462585 EC50 = 24 nM T02506 CYW34A 71519686 IC50 = 3000 nM T02506 C83YJF 71544946 IC50 > 5000 nM T02506 CT9Y5D 71549558 IC50 = 3300 nM T02506 C8ZX0F 71549573 IC50 = 7300 nM T02506 CZ8Y7O 71549829 IC50 = 6100 nM T02506 CPFL57 71549843 IC50 = 17000 nM T02506 CY8SP0 71549969 IC50 > 20000 nM T02506 CX6JR5 71550242 IC50 = 7900 nM T02506 C6WIA2 71550244 IC50 = 6300 nM T02506 CSHT69 71550657 IC50 > 5000 nM T02506 COTM69 71580895 IC50 = 0.3 nM T02506 C8L6YZ 71609799 IC50 = 0.2 nM T02506 CNJD68 71609989 IC50 = 0.1 nM T02506 CB0N4Z 71609990 IC50 = 0.2 nM T02506 C6BDX7 71610523 IC50 = 1.5 nM T02506 COZ7X9 71610524 IC50 = 0.7 nM T02506 CW93GB 71610797 IC50 = 1.4 nM T02506 CPL0O7 71624342 EC50 = 2180 nM T02506 C9S4KZ 71624466 EC50 = 470 nM T02506 CA7F2B 71624467 EC50 = 1910 nM T02506 CGT86N 71624573 EC50 = 120 nM T02506 C1RV0Q 71624574 EC50 = 45 nM T02506 C2CLE1 71624678 EC50 = 1060 nM T02506 CD23NV 71624679 EC50 = 563 nM T02506 C6NZH1 71624682 EC50 = 65900 nM T02506 COK59Y 71624683 EC50 = 1160 nM T02506 CN06AS 71624796 EC50 = 1520 nM T02506 CFW3R0 71624797 EC50 = 439 nM T02506 CT1KP7 71624798 EC50 = 447 nM T02506 C5Y9LF 71624799 EC50 = 101 nM T02506 CN7KA2 71624911 EC50 = 615 nM T02506 CCFP43 71624912 EC50 = 66 nM T02506 C2C0LQ 71624915 EC50 = 485 nM T02506 CSZA43 71625041 EC50 = 387 nM T02506 C2DFZ4 71625042 EC50 = 9 nM T02506 C81GMJ 71625046 EC50 = 3790 nM T02506 CSOI92 71625169 EC50 = 3890 nM T02506 C1PD9I 71625173 EC50 = 944 nM T02506 C1M9GW 71625174 EC50 = 3640 nM T02506 C5XEQ9 71625175 EC50 = 266 nM T02506 C0OY8P 71661130 EC50 = 48360 nM T02506 CM3N9E 71712303 IC50 = 110 nM T02506 CNRU01 71712304 IC50 = 98 nM T02506 C8EY6K 71714518 IC50 = 1279 nM T02506 CLM0A3 71714519 IC50 = 2900 nM T02506 C8JS5K 71746266 EC50 = 0.8 nM T02506 CHDT07 71746268 EC50 = 0.4 nM T02506 C94DQT 71746269 EC50 = 0.4 nM T02506 CL4YX3 71746650 EC50 = 1.1 nM T02506 C56PQM 71746830 EC50 = 1 nM T02506 CUBP37 71765043 IC50 = 248 nM T02506 C1UA2B 71765044 IC50 = 127 nM T02506 CGJ5X4 71812208 IC50 > 5000 nM T02506 CN9M7E 71817803 IC50 = 222 nM T02506 CW36SK 73057389 IC50 = 145 nM T02506 CIS0D4 73057390 IC50 = 92 nM T02506 C7WEA2 73057393 IC50 = 484 nM T02506 C1AUC0 73057394 EC50 = 221 nM T02506 CE58TN 73333597 IC50 = 3100 nM T02506 CY4W5Z 73333703 IC50 = 12700 nM T02506 CSF52H 73333825 IC50 = 3200 nM T02506 C2RLP9 73346567 IC50 = 64908.26 nM T02506 CK3RU8 73347518 IC50 = 29.7 nM T02506 CA60OG 73348058 IC50 < 100000 nM T02506 CPVB67 73348059 IC50 = 64908.26 nM T02506 C4XOW1 73348859 EC50 = 12570 nM T02506 C5DTJ0 73350233 Ki = 190 nM T02506 CY53FM 73351956 EC50 = 8170 nM T02506 C1ZS5U 73352620 IC50 < 100000 nM T02506 CQN6M8 73353409 EC50 = 2550 nM T02506 C0G1IK 73353410 EC50 = 8320 nM T02506 CW6D9R 73354127 IC50 < 100000 nM T02506 CDKC58 73355642 IC50 < 100000 nM T02506 C9WY3B 73386689 EC50 = 15 nM T02506 CB4Q3X 73671443 EC50 = 6.2 nM T02506 CTVC21 73774965 EC50 = 61.5 nM T02506 C96JWC 73774966 EC50 = 5.2 nM T02506 C46ZFX 73775123 EC50 = 13.9 nM T02506 CK46UZ 73775278 EC50 = 5.3 nM T02506 C3L2WC 73775280 EC50 = 717.1 nM T02506 CCA4K2 74222430 EC50 = 0.8 nM T02506 CYGH56 76317236 IC50 = 14 nM T02506 CA9IX6 76328166 IC50 = 151 nM T02506 CP5E2V 76333018 EC50 = 7943.28 nM T02506 CX3T5H 76335417 IC50 = 100000 nM T02506 C0BF2I 76335716 IC50 = 26200 nM T02506 CA0D6H 76336630 EC50 = 31.62 nM T02506 C1B5KS 76336631 EC50 = 10000 nM T02506 C5KQ9A 77105904 IC50 = 0.4 nM T02506 C36YQX 78321756 IC50 = 23 nM T02506 CC90JF 78321758 IC50 = 78 nM T02506 CPH9Y0 78322066 IC50 = 4 nM T02506 CUD9B4 78322070 IC50 = 327 nM T02506 CELW49 78322377 IC50 = 316 nM T02506 CQ4B9L 78322379 IC50 = 31 nM T02506 C32SAW 78322380 IC50 = 647 nM T02506 C3FQG8 78322381 IC50 = 1 nM T02506 CLM34F 78322699 IC50 = 26 nM T02506 CEU36Z 78322700 IC50 = 941 nM T02506 CBHP24 78322701 IC50 = 886 nM T02506 C1G7VK 78322702 IC50 = 1030 nM T02506 CCP63W 78323006 IC50 = 1270 nM T02506 CBUP57 78323007 IC50 = 1823 nM T02506 CQMW35 78323008 IC50 = 26 nM T02506 CN2R0V 78323010 IC50 = 5020 nM T02506 CE09GU 78323328 IC50 = 1 nM T02506 C1MKR2 78323656 IC50 = 6 nM T02506 CG87TA 78323657 IC50 = 1 nM T02506 CNI07G 78323954 IC50 = 1 nM T02506 CY7DO8 78323955 IC50 = 58 nM T02506 C6Y5TP 78323956 IC50 = 40 nM T02506 C74MXP 78324253 IC50 = 55 nM T02506 C96CAJ 78324565 IC50 = 11 nM T02506 CZD3W9 78324876 IC50 = 17 nM T02506 C0ZE4D 78425809 EC50 = 2.1 nM T02506 CF3Q7K 86270891 EC50 = 0.6 nM T02506 C8J1FY 86270985 EC50 = 0.7 nM T02506 CRW92N 86270987 EC50 = 83 nM T02506 CIHS37 86270988 EC50 = 99 nM T02506 C7XPD4 86270989 EC50 = 1.8 nM T02506 CDJN45 86271086 EC50 = 37 nM T02506 C2VJ8M 86271087 EC50 = 7.4 nM T02506 CI9Y8M 86271089 EC50 = 1.7 nM T02506 CG79NV 86271184 EC50 = 17 nM T02506 CIF3C7 86271185 EC50 = 50 nM T02506 CA6PM4 86271186 EC50 = 28 nM T02506 CB5P2N 86271281 EC50 = 15 nM T02506 C8A1OX 86271282 EC50 = 300 nM T02506 CZ3D7B 86271283 EC50 = 90 nM T02506 CM83WK 86271284 EC50 = 12 nM T02506 C47MPR 86271285 EC50 = 190 nM T02506 CV0J7G 86271469 EC50 = 0.8 nM T02506 CA6J1C 86271471 EC50 = 1.1 nM T02506 CV90DA 86271553 EC50 = 1.6 nM T02506 CZ1N5T 86271645 EC50 = 4.2 nM T02506 C5KQ2Z 86271646 EC50 = 1.1 nM T02506 C5U6BO 86271738 EC50 = 5 nM T02506 C95BEZ 86271739 EC50 = 1.5 nM T02506 C1IZH2 86271742 EC50 = 1.9 nM T02506 C13XTI 86271833 EC50 = 0.8 nM T02506 CVQ71C 86271835 EC50 = 4.8 nM T02506 CHVL65 86271924 EC50 = 1.4 nM T02506 CP26ZM 86271925 EC50 = 2.8 nM T02506 CWN65V 86271926 EC50 = 4.1 nM T02506 CNEP10 86345430 IC50 = 1 nM T02506 C31WCG 86346166 IC50 = 0.1 nM T02506 CQRK65 86730685 IC50 = 3400 nM T02506 CTU83L 86763463 IC50 = 15 nM T02506 CB1VC0 86764136 IC50 = 0.4 nM T02506 CUJA92 86764241 IC50 = 0.2 nM T02506 C59GJF 87054925 IC50 = 13 nM T02506 C2U0BG 87055263 IC50 = 0.03 nM T02506 C5JK1L 89042295 IC50 = 112 nM T02506 CJSX36 89619690 IC50 = 0.2 nM T02506 CO07PH 89619977 IC50 = 0.1 nM T02506 C4O8HY 89634497 IC50 = 0.2 nM T02506 CB3I2O 89634514 IC50 = 11 nM T02506 CZH25C 89634609 IC50 = 0.1 nM T02506 CHVM10 89820253 EC50 = 4.3 nM T02506 CY6UE5 89820263 EC50 = 19 nM T02506 CJ0U4Y 89820264 EC50 = 0.3 nM T02506 CT3M7I 89820265 EC50 = 1.5 nM T02506 CMQ93G 90348277 IC50 > 10000 nM T02506 CF53CX 90372168 IC50 = 0.2 nM T02506 CK5F0Y 90372180 IC50 = 124 nM T02506 C5GFU4 90372433 IC50 = 5.4 nM T02506 CS3TR0 90372437 IC50 = 0.3 nM T02506 CVI17J 90372445 IC50 = 4.2 nM T02506 CK5D1A 90395281 IC50 = 17000 nM T02506 CK7MX2 90644079 EC50 = 0.3 nM T02506 C9S3GC 90644080 EC50 = 2.7 nM T02506 CB0QV8 90644081 EC50 = 20 nM T02506 C6YH5U 90644082 IC50 = 3 nM T02506 CEXC10 90644320 EC50 = 16 nM T02506 C1J2TA 90654352 IC50 = 26.2 nM T02506 COG3Q5 91668558 IC50 = 117 nM T02506 CYI89C 91810785 IC50 = 6.5 nM T02506 CU5XG6 102228006 IC50 = 10 nM T02506 CNJH98 102502192 EC50 = 96 nM T02506 C5ZR2C 102502193 EC50 = 61 nM T02506 CMO84S 110730849 IC50 = 204.75 nM T02506 C9FIG4 110730850 IC50 = 3.31 nM T02506 CIUL38 110730851 IC50 = 7.53 nM T02506 C6BDS9 112513964 IC50 = 69.46 nM T02506 C6VH5J 117094740 IC50 = 43 nM T02506 CNK71A 117611174 EC50 = 1.9 nM T02506 CX5FR2 117763076 IC50 = 0.3 nM T02506 CW27MY 118063735 EC50 > 10000 nM T02506 CI4GP9 118097391 EC50 > 10000 nM T02506 CQT2M7 118166573 IC50 = 1030 nM T02506 CU03DL 118166622 IC50 = 0.9 nM T02506 CB10GA 118166666 IC50 = 262 nM T02506 CF6MO1 118166678 IC50 = 7 nM T02506 CL5I0X 118166693 IC50 = 56 nM T02506 CV7ZG9 118166698 IC50 = 7 nM T02506 C7A8UH 118166720 IC50 = 113 nM T02506 CT0PZ7 118166734 IC50 = 0.8 nM T02506 CRTP56 118166740 IC50 = 120 nM T02506 CV2M7R 118166744 IC50 = 110 nM T02506 CH9QA7 118166788 IC50 = 219 nM T02506 CR32JE 118166789 IC50 = 2564 nM T02506 C7FD2S 118166792 IC50 = 112 nM T02506 C08UFT 118166812 IC50 = 1409 nM T02506 C24VKX 118166813 IC50 = 35 nM T02506 C96HPK 118166861 IC50 = 113 nM T02506 C69MNX 118184699 IC50 = 46 nM T02506 CBV6N0 118184700 IC50 = 1174 nM T02506 C06GNI 118184720 IC50 = 43 nM T02506 C7ZJR3 118184730 IC50 = 3 nM T02506 CQH23M 118184731 IC50 = 119 nM T02506 C0INJ8 118184735 IC50 = 15 nM T02506 C29NQM 118184739 IC50 = 5.5 nM T02506 CUG2Z0 118184741 IC50 = 0.6 nM T02506 CF6D0X 118184749 IC50 = 57 nM T02506 CRHI05 118184751 IC50 = 55 nM T02506 C5FC9X 118184760 IC50 = 15 nM T02506 CG69BK 118184761 IC50 = 77 nM T02506 CD1RJ8 118184777 IC50 = 0.4 nM T02506 C1Q8JO 118184782 IC50 = 27 nM T02506 CKLZ47 118184786 IC50 = 1.4 nM T02506 CC2YD0 118184807 IC50 = 207 nM T02506 C4LT7O 118184808 IC50 = 302 nM T02506 CK15YV 118184833 IC50 = 37500 nM T02506 CDK5I7 118184845 IC50 = 12 nM T02506 C4SBX9 118184846 IC50 = 139 nM T02506 CDKC49 118184849 IC50 = 505 nM T02506 C3JIB2 118184854 IC50 = 125 nM T02506 CIML42 118574931 IC50 = 216 nM T02506 CD3CK7 118574963 IC50 = 3 nM T02506 CLS7C1 118707978 Ki > 75000 nM T02506 C9LV0M 118707979 Ki > 75000 nM T02506 C6NIU0 118724546 IC50 = 13000 nM T02506 C3JU5H 118724548 IC50 = 230 nM T02506 C4UB8J 118724549 IC50 = 1100 nM T02506 CE0C6J 118724550 IC50 = 140 nM T02506 C7BRJ0 118724551 IC50 = 150 nM T02506 C5LR2N 118724552 IC50 = 40 nM T02506 CG1OL3 118724553 IC50 = 1470 nM T02506 CCK94J 118724554 IC50 = 18000 nM T02506 CW07TL 118724555 IC50 = 8 nM T02506 COJ81W 118735362 EC50 = 87.8 nM T02506 C8VFT2 118735363 EC50 = 277 nM T02506 CZE92I 118735364 EC50 = 274 nM T02506 CFB1G7 118735365 EC50 = 144 nM T02506 CX4V1E 118735366 EC50 = 1050 nM T02506 CW60ZD 118735367 EC50 = 675 nM T02506 C6ULM1 118735368 EC50 = 265 nM T02506 CE50LC 118735369 EC50 = 384 nM T02506 C6Y2NQ 118735371 EC50 = 653 nM T02506 C93CNO 118735374 EC50 = 290 nM T02506 C4YR6E 118735375 EC50 = 56.5 nM T02506 CS3ZJ8 118735376 EC50 = 176 nM T02506 CV83KA 118735377 EC50 = 3180 nM T02506 CG9RB4 118735379 EC50 = 34.9 nM T02506 CGT60X 118735380 EC50 = 27.1 nM T02506 CY6L8W 118735381 EC50 = 1920 nM T02506 C7VL3P 118737781 IC50 = 17 nM T02506 CQ4P8B 118737782 IC50 = 41 nM T02506 CZG3N7 118737783 IC50 = 5.9 nM T02506 CM14ON 118737784 IC50 = 9 nM T02506 C5XIC2 118737785 IC50 = 4.6 nM T02506 C5JTP6 118737786 IC50 = 1.6 nM T02506 C6V7AD 118737787 IC50 = 3 nM T02506 CJWX60 118737788 IC50 = 178 nM T02506 CC85BI 118737789 IC50 = 11 nM T02506 CES6O7 118737790 IC50 = 1.5 nM T02506 CNK32A 118737791 IC50 = 1 nM T02506 CUM9T0 118737792 IC50 = 256 nM T02506 CVN7J1 118737793 IC50 = 27 nM T02506 CVH7A9 118737794 IC50 = 0.5 nM T02506 CP4Y1L 118737795 IC50 = 25 nM T02506 CVM93U 118737796 IC50 = 9.9 nM T02506 C6N2PZ 118737797 IC50 = 1.3 nM T02506 CJN28K 118737798 IC50 = 7.4 nM T02506 C2XVQ5 118737799 IC50 = 3.2 nM T02506 C0MK1L 118737800 IC50 = 10 nM T02506 CZ8HX6 118737801 IC50 = 280 nM T02506 CT05AI 118737802 IC50 = 360 nM T02506 C6R2NI 118737803 IC50 = 100 nM T02506 CPA95Q 118737804 IC50 = 390 nM T02506 CBYP36 118737805 IC50 = 3600 nM T02506 CR6X9U 118737806 IC50 = 5800 nM T02506 CI53XV 118737807 IC50 = 330 nM T02506 C6E1WC 118737808 IC50 = 100 nM T02506 CIQ57L 118737845 IC50 = 50 nM T02506 CSJE19 118737846 IC50 = 50 nM T02506 C42PSU 118737847 IC50 = 1380 nM T02506 C8UP2N 121226004 IC50 = 55300 nM T02506 CWE9Y5 121241709 IC50 = 1.1 nM T02506 C0WO6T 121409920 IC50 = 0.58 nM T02506 CT0V7C 121409947 IC50 = 0.03 nM T02506 C68EUS 121409965 IC50 = 0.05 nM T02506 CP7N6H 121409995 IC50 = 0.2 nM T02506 C21AIE 121410016 IC50 = 3 nM T02506 CM2C0V 121410025 IC50 = 1 nM T02506 CZ68RS 121410042 IC50 = 0.5 nM T02506 C7CGK4 121410113 IC50 = 0.01 nM T02506 COS47H 121410578 IC50 = 0.07943 nM T02506 C8FN6J 121427080 IC50 = 0.045 nM T02506 CRUN70 121430327 IC50 = 0.5 nM T02506 CG13LX 122178361 IC50 = 4900 nM T02506 CT4Q1B 122178995 EC50 = 113 nM T02506 CVAY18 122178996 EC50 = 1050 nM T02506 CJ3LN0 122180153 IC50 = 53 nM T02506 C29JVK 122180154 IC50 = 3.6 nM T02506 C0TPU3 122180155 IC50 = 11 nM T02506 C8NQV0 122180156 IC50 = 4.8 nM T02506 C17TCM 122180157 IC50 = 210 nM T02506 C7QCB9 122180158 IC50 = 3.4 nM T02506 CRW9F3 122180812 Ki = 59.86 nM T02506 C3UO8M 122180813 EC50 = 1 nM T02506 CJ42OQ 122180814 Ki = 25 nM T02506 CRH37W 122180815 Ki = 56.57 nM T02506 CEW23B 122180816 Ki = 147.62 nM T02506 CBM0N2 122180817 Ki = 111.91 nM T02506 C7E2QD 122180818 Ki = 182.35 nM T02506 CBO5T8 122180819 Ki = 80.52 nM T02506 C3TB4Y 122180820 Ki = 2384.62 nM T02506 C3D4TV 122180821 EC50 = 1160 nM T02506 CC80JD 122180822 Ki = 104.02 nM T02506 CXPG14 122180823 Ki = 81.36 nM T02506 CS4OH2 122180824 Ki = 133.05 nM T02506 CB7MD5 122180825 EC50 = 16 nM T02506 CB51GT 122180826 Ki = 92.26 nM T02506 C1YZ6A 122180827 IC50 = 140 nM T02506 CYCT17 122180828 Ki = 126.02 nM T02506 COM0C9 122180829 Ki = 125.51 nM T02506 CP5ND8 122180830 IC50 = 790 nM T02506 CTPJ86 122180831 IC50 = 640 nM T02506 C4FJ1W 122180832 EC50 = 320 nM T02506 CF71OE 122180833 Ki = 121.57 nM T02506 CL16JS 122180834 Ki = 169.4 nM T02506 CE2A5S 122180835 Ki > 5000 nM T02506 CBC6D3 122181041 Ki > 5000 nM T02506 CP4ZJ2 122181042 Ki = 4428.57 nM T02506 COEZ74 122181043 Ki > 5000 nM T02506 C0EHV1 122181044 Ki > 5000 nM T02506 CA0KZ7 122181045 Ki > 5000 nM T02506 CE4AO3 122181046 EC50 = 1140 nM T02506 C7XP2A 122181047 Ki > 5000 nM T02506 CYD03G 122181048 IC50 = 160 nM T02506 C7QS2U 122183657 IC50 = 35 nM T02506 CF4V1K 122183658 IC50 = 13 nM T02506 C3KTX1 122183659 IC50 > 1000 nM T02506 CWB39X 122183660 IC50 = 620 nM T02506 C6XR8T 122183661 IC50 = 670 nM T02506 C2JPF0 122183662 IC50 > 1000 nM T02506 CH96CM 122183664 IC50 = 110 nM T02506 CBYI87 122183665 IC50 > 1000 nM T02506 CRUD13 122183666 IC50 > 1000 nM T02506 C1ZU3J 122183667 IC50 = 749 nM T02506 CXM1S6 122183668 IC50 = 94 nM T02506 CQ5IZ1 122183669 IC50 > 1000 nM T02506 C8QO1G 122183672 IC50 > 1000 nM T02506 CTX29Y 122183673 IC50 > 1000 nM T02506 CGJU04 122191773 IC50 = 3100 nM T02506 C0CLX7 122191774 IC50 = 24600 nM T02506 CN9C2T 122192181 IC50 = 1174.9 nM T02506 C80TIN 122192182 IC50 = 3715.35 nM T02506 CZG5N9 122192183 IC50 = 39.81 nM T02506 CBE26N 122192184 IC50 = 776.25 nM T02506 CP5ER0 122192185 IC50 = 43.65 nM T02506 CAR2M7 122192186 IC50 = 30.2 nM T02506 CZMK47 122192187 IC50 = 691.83 nM T02506 CCP56N 122192188 IC50 = 69.18 nM T02506 C3KH0N 122192189 IC50 = 97.72 nM T02506 CI8KN0 122192190 IC50 = 6.457 nM T02506 C95FVG 122192191 IC50 = 0.4169 nM T02506 C0T5CD 122620887 IC50 = 0.059 nM T02506 C7PUB4 122621200 IC50 = 0.055 nM T02506 CK08DJ 122621381 IC50 = 0.076 nM T02506 CP17KA 122622110 IC50 = 0.051 nM T02506 C4P9NG 122700657 EC50 = 289 nM T02506 C6CA4O 124088406 EC50 = 99 nM T02506 CNH4A8 124088429 EC50 > 10000 nM T02506 CEK31I 124148318 IC50 = 0.2512 nM T02506 C9QF2H 124222742 IC50 = 34 nM T02506 CF05QT 126480615 IC50 = 4.1 nM T02506 C94TWG 127025760 EC50 = 0.22 nM T02506 CEN47V 127029860 IC50 = 34.5 nM T02506 CCK36V 127029882 IC50 > 40000 nM T02506 CFY1P0 127029884 IC50 > 2000 nM T02506 C4M8QN 127030254 IC50 = 0.8 nM T02506 CCD7S3 127030255 IC50 = 0.4 nM T02506 CJQ73M 127030543 IC50 = 36 nM T02506 CQPR75 127030544 IC50 = 0.96 nM T02506 C3AFS4 127030545 IC50 = 3.981 nM T02506 CN5XW9 127030559 IC50 = 590 nM T02506 C47AYI 127030560 IC50 = 960 nM T02506 CZG9X5 127030821 IC50 = 82 nM T02506 CLDC46 127031152 IC50 > 37000 nM T02506 C60SMC 127031153 IC50 > 12000 nM T02506 CX4W7N 127031748 IC50 = 12.4 nM T02506 C1NYI0 127031749 IC50 = 81 nM T02506 C6W1YO 127032311 IC50 = 1.2 nM T02506 C4BXE0 127032365 IC50 = 1.7 nM T02506 CHAY10 127032366 IC50 = 1.6 nM T02506 CSN4B7 127032367 IC50 = 7.5 nM T02506 C2SGB4 127032368 IC50 = 1.3 nM T02506 CU0XT5 127032369 IC50 = 0.69 nM T02506 CR24LG 127032671 IC50 = 2.2 nM T02506 C2J4VF 127033264 IC50 = 5.8 nM T02506 CL7R1I 127033595 IC50 = 160 nM T02506 C39DUH 127033596 IC50 = 0.4 nM T02506 C7ZMR6 127033597 IC50 = 1.3 nM T02506 C9D2LE 127033598 IC50 = 0.25 nM T02506 C74SAW 127033892 IC50 = 22 nM T02506 CSV67L 127033893 IC50 = 31.9 nM T02506 C3QCS2 127033894 IC50 = 7.7 nM T02506 C3SR7L 127033895 IC50 = 27.1 nM T02506 CFI4S3 127033896 IC50 = 48.4 nM T02506 CF70TI 127034151 IC50 = 42 nM T02506 C12NMV 127034152 IC50 = 11 nM T02506 CLR2J7 127034153 IC50 = 1.3 nM T02506 CJK82T 127034154 IC50 = 5.5 nM T02506 C6HEU2 127034384 IC50 = 33.3 nM T02506 C0ZNT8 127034418 IC50 = 7 nM T02506 CEO3L9 127034419 IC50 = 170 nM T02506 CC6FD8 127034721 IC50 = 1060 nM T02506 C4EH3T 127034722 IC50 = 210 nM T02506 C2YXR7 127034902 IC50 = 2100 nM T02506 C9ZF0D 127035369 IC50 = 50 nM T02506 CLYC28 127038229 EC50 = 0.2 nM T02506 CUI43M 127041633 EC50 = 121 nM T02506 C1JEB2 127041634 EC50 = 436.2 nM T02506 CFB6K2 127042277 EC50 = 1 nM T02506 CWX5L7 127042278 EC50 = 58.7 nM T02506 C3G5TE 127042279 EC50 = 76.1 nM T02506 C0ZWQ9 127042604 EC50 = 30.6 nM T02506 C6JMT9 127042633 EC50 = 36.8 nM T02506 CEQ91U 127042898 EC50 = 18.5 nM T02506 CA0J4Q 127042930 EC50 = 33.4 nM T02506 CYU8Z5 127043892 IC50 = 18700 nM T02506 CHL5V4 127044059 IC50 = 17700 nM T02506 CV0Q2X 127044060 IC50 = 24900 nM T02506 C9S8CB 127044061 IC50 > 100000 nM T02506 C3SMP8 127045121 IC50 = 3400 nM T02506 CS04DH 127045122 IC50 = 19800 nM T02506 C5HFJ1 127045123 IC50 = 10600 nM T02506 C38BJS 127045271 IC50 > 100000 nM T02506 CF8R9C 127045272 IC50 = 35200 nM T02506 CSQ06E 127045273 IC50 = 6700 nM T02506 CC6W0E 127045274 IC50 = 7200 nM T02506 C9O4RK 127045434 IC50 = 23300 nM T02506 C8PZU3 127045576 IC50 = 39400 nM T02506 CQT56U 127045577 IC50 = 39800 nM T02506 CXK2T9 127045578 IC50 = 40300 nM T02506 CZ6O4S 127045579 IC50 = 38300 nM T02506 CT1Y6M 127049191 IC50 = 40 nM T02506 C24TMQ 127049192 IC50 = 0.09 nM T02506 C7B2GI 127049193 IC50 = 28 nM T02506 C3Q9UY 127049194 IC50 = 11 nM T02506 CZS07N 127049269 IC50 = 574 nM T02506 CLZR97 127049518 IC50 = 1.8 nM T02506 C4ITS1 127050198 IC50 = 380 nM T02506 CQ76OF 127050449 IC50 = 49 nM T02506 C2REL0 127051417 IC50 = 436 nM T02506 CBF64U 127051803 IC50 = 9 nM T02506 C12WOQ 129137247 EC50 = 72.1 nM T02506 CJB4M3 129137266 EC50 = 11036 nM T02506 CJ1N2M 129137280 EC50 = 212.9 nM T02506 CH42QX 129137285 EC50 = 1711 nM T02506 CZSB45 129205486 Ki = 0.65 nM T02506 CT61ZX 129205487 EC50 = 1.1 nM T02506 CV72WR 129205492 Ki = 0.5 nM T02506 CLRO76 129205499 EC50 = 0.07 nM T02506 C6G7VA 129205523 EC50 = 0.65 nM T02506 C1P3FN 129205616 EC50 = 0.24 nM T02506 C3OP0R 130232322 IC50 = 0.2 nM T02506 CG7T9C 130232326 EC50 = 0.2 nM T02506 CD1K0J 130232334 EC50 = 0.7 nM T02506 C75HQC 130232370 EC50 = 8 nM T02506 C1QY3W 130232392 IC50 = 67 nM T02506 C1EC2X 130232400 EC50 = 0.5 nM T02506 CO9A4K 130232401 EC50 = 1.5 nM T02506 CX1U6G 130232404 EC50 = 0.2 nM T02506 C70GWU 130232413 EC50 = 0.7 nM T02506 CRYS10 130232754 EC50 = 0.9 nM T02506 CG8WO3 130232762 IC50 = 0.2 nM T02506 CMX1V2 130232769 EC50 = 2 nM T02506 CP48SA 130232781 EC50 = 0.3 nM T02506 CR4D5M 130232807 EC50 = 0.5 nM T02506 C9GK1L 130232819 EC50 = 0.2 nM T02506 C3J5LN 130232873 EC50 = 1 nM T02506 C9JL4N 130232895 EC50 = 0.5 nM T02506 CI54NM 130232938 EC50 = 3 nM T02506 CF64WI 130232950 IC50 = 0.2 nM T02506 C57ASV 130232954 EC50 = 0.5 nM T02506 COJP50 130233149 EC50 = 2 nM T02506 CJ3UG9 130233175 IC50 = 38 nM T02506 CGZP38 130233179 IC50 = 0.7 nM T02506 C01ZBV 130233184 EC50 = 8 nM T02506 CEGJ04 130233196 EC50 = 0.3 nM T02506 CH5FI9 130233199 EC50 = 0.4 nM T02506 CKAC59 130233229 IC50 = 0.3 nM T02506 CD81EO 130233396 EC50 = 0.7 nM T02506 CN4RF6 132019596 IC50 = 0.3981 nM T02506 C0J4PZ 132046120 IC50 = 0.3981 nM T02506 CFUG87 132046174 IC50 = 0.631 nM T02506 CE9BL3 132046817 IC50 = 1 nM T02506 C32MHI 132046819 IC50 = 0.1995 nM T02506 CW8CI4 132046902 IC50 = 2.512 nM T02506 C5Y3MB 132502976 IC50 = 12 nM T02506 C79GMJ 132578496 IC50 > 10000 nM T02506 CWQK97 134130451 IC50 = 210 nM T02506 C74WMB 134133952 IC50 = 97 nM T02506 C2URL4 134134246 IC50 = 990 nM T02506 CD7NA5 134138492 IC50 = 2000 nM T02506 CCVJ27 134141761 IC50 = 86 nM T02506 CN7GJ2 134143539 IC50 > 10000 nM T02506 CP04WC 134144077 IC50 = 1700 nM T02506 CQO2G7 134148719 IC50 > 10000 nM T02506 CM8NP0 134149281 IC50 = 553 nM T02506 CFBX89 134149623 IC50 = 224 nM T02506 CYG76M 134150509 IC50 = 3340 nM T02506 C89SMK 134152807 IC50 > 10000 nM T02506 C1O0IW 134153257 IC50 > 10000 nM T02506 CK1BE9 134155077 EC50 = 451.2 nM T02506 C0Z4OD 134155524 IC50 = 875 nM T02506 C2BK3Z 134155779 EC50 = 164.1 nM T02506 C58OUX 134155994 IC50 = 20 nM T02506 CE08RT 134521164 EC50 = 0.3 nM T02506 CX53IF 134610856 IC50 = 10 nM T02506 C31BDG 134822336 IC50 = 195 nM T02506 C1G9FD 135348960 EC50 > 10000 nM T02506 C42PVJ 135400902 IC50 = 65 nM T02506 CL51KF 135400937 IC50 = 49 nM T02506 CBRN70 135400938 IC50 = 33 nM T02506 CY2GJ3 135401184 IC50 = 1500 nM T02506 CLX32H 135409570 Ki = 51 nM T02506 C6S5RV 135409748 IC50 = 246 nM T02506 CY39LP 135409961 IC50 = 1750 nM T02506 CO95DR 135409966 IC50 = 474 nM T02506 CMQE75 135412817 IC50 = 183 nM T02506 C1VWL3 135415992 IC50 = 7827 nM T02506 CPC1Q3 135421346 Ki = 25.12 nM T02506 CLN16H 135423261 IC50 = 47 nM T02506 C3BU7D 135423323 Ki = 7.943 nM T02506 CCRX48 135424620 IC50 = 98 nM T02506 CP9JN3 135424801 IC50 = 27569 nM T02506 C0KIP8 135425149 IC50 = 1753 nM T02506 CV2WX8 135428120 IC50 = 3 nM T02506 CXNV83 135430308 IC50 = 411 nM T02506 C30QWY 135430315 IC50 = 455 nM T02506 CK2ZF0 135431815 IC50 > 5000 nM T02506 CYJ7R0 135432882 IC50 = 8.5 nM T02506 CWCV13 135433141 Ki = 450 nM T02506 CA1MC6 135433906 IC50 = 30 nM T02506 CCI27T 135433989 IC50 = 196 nM T02506 CW7MZ8 135436561 IC50 > 5000 nM T02506 CAY0S9 135436566 IC50 = 4820 nM T02506 CCR8P7 135438141 IC50 = 475 nM T02506 C43PRB 135438183 EC50 = 3070 nM T02506 CC29NQ 135438201 IC50 = 463 nM T02506 CDA4B8 135438473 IC50 = 2260 nM T02506 CUXH34 135440385 Ki = 15.85 nM T02506 CBGO63 135443283 IC50 = 555 nM T02506 C8VWH0 135443287 IC50 = 5000 nM T02506 CX1T4W 135443301 IC50 = 1210 nM T02506 C21VTE 135445165 Ki = 125.89 nM T02506 CE50DW 135445365 IC50 = 1010 nM T02506 C60OGT 135445374 IC50 = 1340 nM T02506 CVM0P7 135446139 IC50 = 2854 nM T02506 CTD6A7 135449071 IC50 = 511 nM T02506 C78GFC 135454762 IC50 = 622 nM T02506 C9GZ1Q 135454811 IC50 = 1815 nM T02506 CEQ5F4 135457031 IC50 > 5000 nM T02506 C9BVI8 135457325 IC50 = 260 nM T02506 C2O1MP 135457889 Ki = 26 nM T02506 C1Z4BN 135458008 IC50 = 13 nM T02506 CCVE26 135458128 IC50 = 1309 nM T02506 CXU79B 135458129 IC50 = 3138 nM T02506 CY8U6E 135459005 IC50 > 100000 nM T02506 CHU54B 135461939 IC50 = 9620 nM T02506 CEB1W8 135471179 IC50 > 5000 nM T02506 CPO9D1 135477943 IC50 = 283 nM T02506 C17LIP 135481146 IC50 = 1435 nM T02506 C4O7RZ 135481158 IC50 > 10000 nM T02506 C8SE4C 135483639 IC50 = 2975 nM T02506 C6V1JZ 135483640 IC50 = 44 nM T02506 C6DI2R 135483660 IC50 = 1036 nM T02506 C0WP9D 135486163 EC50 = 901 nM T02506 CH9OV8 135487481 IC50 = 3080 nM T02506 CFO4V6 135489088 IC50 = 1047 nM T02506 CQ91HA 135489089 IC50 = 385 nM T02506 CAU4W8 135489212 Ki = 3162.28 nM T02506 CXY1Z2 135492323 IC50 = 431 nM T02506 CL5WG2 135492495 EC50 = 140 nM T02506 CMB9Z7 135493223 IC50 = 1813 nM T02506 CL20ZX 135494500 IC50 = 410 nM T02506 CTN2D6 135495080 IC50 = 227 nM T02506 CX3O9M 135495087 IC50 = 4040 nM T02506 CFDO01 135496191 IC50 = 1870 nM T02506 CB9Q3X 135496242 Ki = 10 nM T02506 CMK68Q 135497123 IC50 = 803 nM T02506 C90ZNW 135497128 Ki = 10 nM T02506 C2O8MY 135499764 IC50 = 717 nM T02506 CI09WX 135499787 IC50 = 3370 nM T02506 CE1D4V 135499837 IC50 = 2668 nM T02506 C3N9DF 135499972 IC50 = 443 nM T02506 CZ5Y9F 135500018 IC50 = 50 nM T02506 C25GWU 135500024 IC50 = 360 nM T02506 CRYW41 135502641 IC50 = 1100 nM T02506 C1RW9U 135503521 IC50 = 68 nM T02506 COF53G 135507181 Ki = 160 nM T02506 C67JAI 135507439 IC50 = 20 nM T02506 CPZ29O 135508382 IC50 = 163 nM T02506 C2ME7Q 135508383 IC50 = 809 nM T02506 C9GM1V 135508397 IC50 = 1980 nM T02506 CHO9X5 135508451 IC50 = 15 nM T02506 CFMN96 135511852 EC50 = 59 nM T02506 CJ60KF 135511863 EC50 = 1217 nM T02506 C7PZI5 135511869 IC50 = 2636 nM T02506 C9DZ7C 135511925 IC50 = 96 nM T02506 C67GSY 135511929 EC50 = 4790 nM T02506 CR7X1H 135511945 EC50 = 149 nM T02506 C61NSW 135514474 Ki = 100 nM T02506 CV6B8P 135515561 Ki = 20 nM T02506 C4XD9K 135516685 IC50 = 50 nM T02506 CGM5C6 135516694 IC50 = 6 nM T02506 CZKC69 135518123 IC50 = 24 nM T02506 CBPO32 135518124 IC50 = 1727 nM T02506 CVTD54 135518270 IC50 = 783 nM T02506 C3S5MX 135518313 IC50 = 559 nM T02506 CH6G0Q 135519304 IC50 = 4068 nM T02506 C3P8LZ 135519309 IC50 = 264 nM T02506 CU5J8M 135520120 IC50 = 48473 nM T02506 CR03JM 135522279 IC50 = 2638 nM T02506 C1OBI2 135524469 IC50 = 210 nM T02506 CNFZ03 135524510 EC50 = 549 nM T02506 CVX9H3 135524526 IC50 = 22 nM T02506 CMIE65 135524868 IC50 > 5000 nM T02506 C7TYU2 135524871 IC50 = 1030 nM T02506 C35TQU 135524884 IC50 = 59 nM T02506 CC46RN 135524945 Ki = 1584.89 nM T02506 CFQW27 135526994 IC50 = 273 nM T02506 CSZ1H7 135527005 EC50 = 140 nM T02506 CRKD27 135529495 Ki = 180 nM T02506 CQ0ZX7 135529496 Ki = 1260 nM T02506 CX1J8D 135535917 IC50 = 161 nM T02506 C15FTQ 135538030 IC50 = 138 nM T02506 CUCN57 135540445 IC50 = 1116 nM T02506 C84ZFX 135540483 IC50 = 31 nM T02506 CIKD94 135545359 IC50 = 249 nM T02506 C7X2CE 135547714 Ki = 7 nM T02506 CK7UM1 135547715 Ki = 47 nM T02506 C34JMK 135571931 IC50 > 100000 nM T02506 C4ODC2 135678114 Ki = 3333 nM T02506 CM0LN8 135817419 IC50 = 1 nM T02506 CSO3C1 135857090 IC50 = 1000 nM T02506 CED1L7 135871534 IC50 < 100000 nM T02506 CSY5I0 135871535 IC50 < 100000 nM T02506 CDJ1L6 135914665 EC50 > 100000 nM T02506 CALV45 135976649 Ki = 4200 nM T02506 CMJ41H 135987657 Ki = 490 nM T02506 CO0UC2 135987660 Ki = 2000 nM T02506 CP96SU 135987662 Ki = 210 nM T02506 C3I8VE 135987663 Ki = 650 nM T02506 CDG17Y 135987664 Ki > 3000 nM T02506 C9ABZ6 135987665 Ki = 130 nM T02506 C7GU8Q 135987666 Ki = 830 nM T02506 C4G1DL 135987668 Ki = 660 nM T02506 CIG6T5 135987670 Ki = 380 nM T02506 C1TV3R 135987671 Ki = 620 nM T02506 CSB76X 135987672 Ki = 70 nM T02506 C5B8SX 136002646 IC50 = 5100 nM T02506 C98FXW 136046127 EC50 = 3 nM T02506 CUN8F1 136046128 EC50 = 7 nM T02506 CX2KM3 136046129 EC50 = 5 nM T02506 CSOR78 136046131 EC50 = 1 nM T02506 CB1L2D 136046132 EC50 = 10 nM T02506 CQTA24 136046133 EC50 = 2 nM T02506 CB6YN3 136046134 EC50 = 23 nM T02506 CJ7AO4 136046135 EC50 = 2 nM T02506 C68OIK 136046136 EC50 = 1 nM T02506 CQ7K2A 136046137 EC50 = 14 nM T02506 CSCP10 136046138 EC50 = 7 nM T02506 C9LMN8 136046140 EC50 = 14 nM T02506 CJSU38 136046141 EC50 = 16 nM T02506 CU18VS 136046142 EC50 = 0.1 nM T02506 C5ORA9 136046143 EC50 = 15 nM T02506 CFGU03 136046144 EC50 = 4 nM T02506 CJ8X1O 136046145 EC50 = 57 nM T02506 C4P2BT 136046146 EC50 = 10 nM T02506 CXTR87 136046147 EC50 = 9 nM T02506 C9BI5M 136046148 EC50 = 7 nM T02506 CAH5S3 136046149 EC50 = 17 nM T02506 C0YZM4 136048726 IC50 = 376 nM T02506 CMI3Z2 136048727 IC50 = 196 nM T02506 C1BE8P 136048728 IC50 = 539 nM T02506 CRVT63 136048730 IC50 = 4652 nM T02506 CZG20O 136053633 EC50 = 64 nM T02506 CJC8N5 136053634 EC50 = 6900 nM T02506 CV3TP6 136053635 EC50 = 1400 nM T02506 CNW6H0 136053636 EC50 = 1700 nM T02506 C5WTV7 136053637 EC50 = 170 nM T02506 CRBK35 136053638 EC50 = 170 nM T02506 CRV6U5 136053639 EC50 = 46 nM T02506 C54YLG 136053640 EC50 = 12000 nM T02506 CCB5P6 136053641 EC50 = 1800 nM T02506 CO60LF 136053642 EC50 = 2000 nM T02506 CB54HV 136053643 EC50 = 900 nM T02506 CRA6C4 136053644 EC50 = 3100 nM T02506 CM35UY 136180341 EC50 = 29.3 nM T02506 CXP07U 136180342 EC50 = 194 nM T02506 CO79XD 136213601 IC50 = 7750 nM T02506 CR0ND2 136213603 IC50 = 1 nM T02506 CM9D8R 136213604 IC50 = 3 nM T02506 CVY5F4 136244610 IC50 < 100000 nM T02506 C38YOM 136260557 IC50 < 100000 nM T02506 C5GWA9 136497898 IC50 = 219 nM T02506 CKJ2F4 137175229 EC50 = 75 nM T02506 CC1XZ2 137175230 EC50 = 46 nM T02506 CM6EA1 137175231 EC50 = 77 nM T02506 CGH34U 137194225 EC50 = 0.2 nM T02506 C4HRL1 137503296 IC50 = 0.955 nM T02506 C4X2UQ 137503299 IC50 = 1.23 nM T02506 C5O4IG 137503303 IC50 = 1.023 nM T02506 C5IMN2 137503342 IC50 = 2.7 nM T02506 CC98EO 137503344 IC50 = 1.445 nM T02506 CZ90FS 137503669 IC50 = 1.413 nM T02506 CNXJ86 137628681 IC50 = 1943 nM T02506 CG79XQ 137631712 IC50 = 3510 nM T02506 CC64EG 137633461 Ki = 1.4 nM T02506 C2B3GJ 137634109 Ki = 0.13 nM T02506 CT03AC 137634796 Ki = 0.37 nM T02506 CMN0U2 137635165 IC50 = 63.2 nM T02506 CZ3V1F 137635423 Ki = 0.43 nM T02506 CIAM46 137637216 Ki = 0.18 nM T02506 C8OJ0I 137638372 Ki = 1.1 nM T02506 C2N3FX 137638822 IC50 = 1681 nM T02506 CP2VE3 137638954 IC50 = 2650 nM T02506 C85UAK 137639567 Ki = 0.35 nM T02506 CJV72U 137639609 Ki = 7.1 nM T02506 C9T6JB 137639849 IC50 = 6640 nM T02506 C32YMC 137640489 Ki = 0.57 nM T02506 CF8DG7 137640807 IC50 = 219 nM T02506 CLTS71 137641590 IC50 = 169 nM T02506 C8HP3M 137642810 Ki = 0.45 nM T02506 CRS0C8 137643006 IC50 = 294 nM T02506 CV5HA4 137643922 IC50 = 664 nM T02506 C5C9WQ 137645325 Ki = 3.3 nM T02506 CBY5H6 137645495 Ki = 0.71 nM T02506 C5Y2FO 137645971 IC50 = 10000 nM T02506 C2G3VI 137646525 Ki = 0.4 nM T02506 CHT21E 137646826 IC50 = 27 nM T02506 C9CWP1 137647667 Ki = 0.74 nM T02506 CX0JA8 137647962 Ki = 0.32 nM T02506 C5M7SV 137648055 IC50 = 158 nM T02506 CWP5O2 137649257 EC50 = 432 nM T02506 C8FVM1 137649725 IC50 = 1238 nM T02506 CE7K8L 137649825 Ki = 0.43 nM T02506 CNI49S 137650614 Ki = 0.37 nM T02506 C3O8KX 137651054 IC50 = 271 nM T02506 CR72HJ 137652183 Ki = 0.27 nM T02506 C2FZG3 137652281 IC50 = 1138 nM T02506 C8TR4J 137652311 IC50 > 10000 nM T02506 CWJ40L 137652508 IC50 = 154 nM T02506 CMR9Z4 137652975 IC50 = 1083 nM T02506 C1AS5K 137653286 IC50 = 9390 nM T02506 C57LME 137654397 Ki = 1.33 nM T02506 CMOA79 137656420 Ki = 0.36 nM T02506 CUPZ80 137657526 IC50 = 1654 nM T02506 C9LR5G 137658509 IC50 = 36 nM T02506 C7XP9V 137659010 Ki = 0.71 nM T02506 C40IML 137659097 Ki = 0.65 nM T02506 C1PE7V 137659936 Ki = 0.38 nM T02506 CN0SZ4 137660238 Ki = 0.37 nM T02506 C9FA3U 137660578 Ki = 1.7 nM T02506 CSQH43 137661589 IC50 = 225 nM T02506 CZ03SK 137661821 Ki = 0.71 nM T02506 CVY1M4 137662307 Ki = 1.8 nM T02506 CM3UF7 137700779 IC50 > 20000 nM T02506 CF1VR5 138693144 IC50 = 0.8 nM T02506 CC3E0R 138693215 IC50 = 0.5 nM T02506 C4U5PM 138693278 IC50 = 0.5 nM T02506 C01WKT 138693350 IC50 = 0.5 nM T02506 CPV1E4 138693568 IC50 = 0.6 nM T02506 CZ9E1A 139391843 IC50 = 2.1 nM T02506 CB0E1Y 139392008 IC50 = 8.128 nM T02506 CEO3I4 139392056 IC50 = 10.47 nM T02506 CA3I7J 139408644 IC50 = 5.129 nM T02506 CWKI95 139408668 IC50 = 12 nM T02506 C0K2JE 139408674 IC50 = 0.257 nM T02506 CPH0L4 139408675 IC50 = 1.905 nM T02506 CSXU49 139408681 IC50 = 3.02 nM T02506 CYS5L7 139408845 IC50 = 5.888 nM T02506 CMH90D 139408877 IC50 = 1.023 nM T02506 C6FJE2 139408939 IC50 = 5.2 nM T02506 CW2C4Z 139408951 IC50 = 0.5 nM T02506 CF8LN1 139582020 IC50 = 0.7943 nM T02506 CV26PQ 139582021 IC50 = 0.3981 nM T02506 CO05VM 145949224 IC50 = 539.18 nM T02506 CVC0B4 145950353 IC50 > 10000 nM T02506 CS05YB 145950468 IC50 = 5970 nM T02506 CZNX35 145951019 IC50 = 78 nM T02506 C4T0UE 145951407 IC50 > 10000 nM T02506 CHC8A3 145951614 IC50 > 10000 nM T02506 CWI7X0 145951633 IC50 = 168 nM T02506 CX9LI1 145951641 IC50 = 6430 nM T02506 CGSQ41 145952207 IC50 = 46.88 nM T02506 CRS3V5 145952243 IC50 > 10000 nM T02506 CGT02H 145953052 IC50 = 73.61 nM T02506 CJ86FH 145953150 IC50 = 8430 nM T02506 CG0YF8 145953184 IC50 = 80.36 nM T02506 C8WVA0 145953503 IC50 = 13200 nM T02506 CKP95X 145953707 IC50 > 10000 nM T02506 C97OLA 145953737 IC50 = 387.37 nM T02506 C2ZX1U 145953877 IC50 = 191.69 nM T02506 C65TWJ 145953883 IC50 > 10000 nM T02506 CCK17E 145953908 IC50 = 2190 nM T02506 CC7X6N 145953909 IC50 = 6870 nM T02506 CQ6N9J 145953976 IC50 = 3550 nM T02506 C7AUH9 145953977 IC50 > 10000 nM T02506 CX3BS8 145954021 IC50 = 6620 nM T02506 C8RA6E 145954397 IC50 = 4.9 nM T02506 CTV6X8 145954466 IC50 = 87 nM T02506 C3XOI2 145954572 IC50 = 3820 nM T02506 COK71C 145954893 IC50 = 6840 nM T02506 C0JNE2 145955665 IC50 = 4530 nM T02506 C6DK3T 145956091 IC50 = 16200 nM T02506 CM4W3N 145956205 IC50 = 259.16 nM T02506 CP69IC 145956222 IC50 = 60400 nM T02506 C1D4QT 145956476 IC50 = 4370 nM T02506 CN71VU 145956504 IC50 = 9420 nM T02506 CRN8U6 145956586 IC50 = 201.81 nM T02506 CO18XW 145957375 IC50 = 6430 nM T02506 CW21YS 145957522 IC50 = 78 nM T02506 C2Q5GH 145957892 IC50 = 33.13 nM T02506 CXU20C 145958661 IC50 = 76.73 nM T02506 CR58VX 145959073 IC50 = 300.43 nM T02506 C5IFM0 145959340 IC50 > 10000 nM T02506 CT0QR2 145959503 IC50 = 29400 nM T02506 CS0G2T 145959695 IC50 = 7790 nM T02506 C1WZ5V 145959741 IC50 = 8210 nM T02506 C5KOI6 145959948 IC50 > 200000 nM T02506 C7RK8L 145960186 IC50 = 4.9 nM T02506 C2X7DZ 145960328 IC50 = 7960 nM T02506 CKBW57 145960786 IC50 = 20 nM T02506 CKN29E 145961426 IC50 = 2620 nM T02506 C3U4RJ 145961651 IC50 > 10000 nM T02506 CCF02H 145964530 IC50 = 4100 nM T02506 C56SHA 145964597 IC50 = 4700 nM T02506 CMG6W2 145964616 Ki = 107.38 nM T02506 CVJ7L6 145964633 Ki = 62.1 nM T02506 C8QI0U 145965134 Ki = 51.32 nM T02506 CHF39D 145965184 IC50 = 55000 nM T02506 C9A3UM 145965217 IC50 = 2 nM T02506 C5H8EZ 145965425 IC50 = 1700 nM T02506 C2T3PU 145965787 IC50 = 0.5 nM T02506 CM9LG0 145965903 Ki = 168.6 nM T02506 C8K1WV 145965925 Ki = 153.07 nM T02506 CA6CZ4 145966389 IC50 = 19 nM T02506 CS9MD6 145966668 Ki = 129.74 nM T02506 C0WG5H 145966819 Ki = 498.57 nM T02506 CU4MD5 145967018 IC50 = 26640 nM T02506 CE4S7F 145967279 IC50 = 48 nM T02506 CNJO46 145967622 IC50 = 57 nM T02506 C80AGW 145967704 IC50 = 59 nM T02506 CB68HI 145967819 IC50 = 22440 nM T02506 C8KNI7 145967847 IC50 = 429 nM T02506 C8H3YV 145968201 IC50 = 71.6 nM T02506 C8VQ5G 145968272 IC50 > 10000 nM T02506 C1S0TJ 145968278 IC50 = 4.1 nM T02506 CXN86W 145968289 IC50 = 349 nM T02506 CE1WK0 145968307 IC50 = 634 nM T02506 C8BF1J 145968369 IC50 = 11.7 nM T02506 CRUO57 145968523 IC50 = 147 nM T02506 C2CE4P 145968537 IC50 = 104 nM T02506 CD86FU 145968562 IC50 = 1023 nM T02506 CY78XO 145968786 IC50 = 1040 nM T02506 C2DNL3 145968920 IC50 = 482300 nM T02506 CT8R7I 145968943 Ki = 249.29 nM T02506 CL6IQ4 145969020 IC50 = 613 nM T02506 C40OKG 145969029 IC50 > 10000 nM T02506 CEQ15L 145969388 IC50 = 60780 nM T02506 CY0VA4 145969440 IC50 = 14 nM T02506 C86AEM 145969473 IC50 = 1129 nM T02506 CO75XN 145969585 IC50 = 14 nM T02506 CEY2I5 145969791 IC50 = 21 nM T02506 C7PQH3 145969854 IC50 = 49 nM T02506 CXY0E1 145970107 IC50 = 74 nM T02506 CW1D3A 145970135 IC50 > 10000 nM T02506 C93BQD 145970491 IC50 = 61080 nM T02506 CVY9Q7 145971019 IC50 = 587190 nM T02506 CH0X7P 145971353 IC50 = 355790 nM T02506 CVW6D7 145972047 Ki = 240.69 nM T02506 C4KJX2 145972317 Ki = 634.55 nM T02506 CAVN67 145972459 IC50 = 4270 nM T02506 CLJ4Y7 145972474 IC50 > 10000 nM T02506 CQ47XM 145972475 IC50 > 10000 nM T02506 C1QF2L 145972690 IC50 = 2.4 nM T02506 CDQ7E0 145972963 Ki > 10000 nM T02506 C4OF2V 145973074 IC50 = 5 nM T02506 C5TP2F 145973118 IC50 = 400 nM T02506 CI6T9M 145973161 IC50 = 40 nM T02506 C37FBS 145973441 Ki = 251.08 nM T02506 CFKW97 145973654 IC50 = 18410 nM T02506 C3AZ4O 145973866 Ki = 29.7 nM T02506 CXZS64 145974009 IC50 = 10 nM T02506 CWC19X 145974551 IC50 > 10000 nM T02506 CJ62QA 145974791 IC50 = 8960 nM T02506 CQZ7D8 145975059 Ki = 40.77 nM T02506 CM01NE 145975361 IC50 = 2 nM T02506 C5V2AD 145975958 IC50 = 16550 nM T02506 C5MJ9W 145975973 IC50 = 3860 nM T02506 CE5N1B 145976228 IC50 = 54 nM T02506 C4Q9KI 145976280 IC50 = 61 nM T02506 CR0ON9 145976505 IC50 = 51190 nM T02506 C8DS5Q 145976853 Ki = 149.15 nM T02506 C4DPO7 145976892 EC50 = 4 nM T02506 CRJU43 145976968 Ki = 53.28 nM T02506 CO70FX 145977155 IC50 = 9270 nM T02506 C7IL3R 145977161 Ki = 10.51 nM T02506 CE75OD 145977494 EC50 = 18 nM T02506 CVX45W 145977605 IC50 = 62 nM T02506 C9MG6O 145977673 Ki = 43.03 nM T02506 C98CHS 145977976 IC50 = 5200 nM T02506 CKQ5C2 145978265 EC50 = 2 nM T02506 CS0N8E 145978277 IC50 = 3 nM T02506 C0D9ES 145978643 IC50 = 0.4 nM T02506 C43SYL 145978903 IC50 = 974 nM T02506 C1AJL5 145979357 EC50 = 116 nM T02506 CCBN24 145979638 IC50 = 415 nM T02506 CE80KP 145980527 IC50 = 874 nM T02506 CJ5U0Y 145980901 EC50 = 136 nM T02506 CLJ3S7 145981530 IC50 = 13 nM T02506 CVC58M 145981549 EC50 = 911 nM T02506 C21SIT 145981553 IC50 = 69 nM T02506 CSM61H 145981867 IC50 = 1589 nM T02506 C7UH4A 145982555 IC50 = 5130 nM T02506 C9KR5H 145982571 IC50 = 2170 nM T02506 CY08OG 145982591 IC50 = 1120 nM T02506 C8UZV2 145982754 IC50 = 3420 nM T02506 CRT9I3 145982975 IC50 = 800 nM T02506 C10XYG 145983072 IC50 = 1200 nM T02506 CNOG85 145983259 IC50 = 1940 nM T02506 C0O1NY 145983278 IC50 = 2860 nM T02506 CCRI70 145983336 Ki = 25 nM T02506 CD69JB 145983784 IC50 = 10000 nM T02506 C05MBI 145983837 IC50 = 390 nM T02506 CP27UK 145983884 Ki = 11 nM T02506 CYZO43 145984038 Ki = 185 nM T02506 CYUD47 145984188 IC50 = 220 nM T02506 CVJY47 145984216 Ki = 0.07 nM T02506 CVH6Y9 145984234 IC50 = 5960 nM T02506 CY79IW 145984263 IC50 = 760 nM T02506 CQ9A0N 145984791 IC50 = 4740 nM T02506 CDM05I 145985073 IC50 = 80 nM T02506 C0O2AR 145985081 IC50 = 89 nM T02506 CEF7W4 145985090 IC50 = 1640 nM T02506 C9MV2L 145985198 IC50 = 820 nM T02506 CC3U1S 145985468 IC50 = 6220 nM T02506 CO50ZW 145985605 Ki = 1541 nM T02506 C3O4HE 145985821 Ki = 6.9 nM T02506 C31MIF 145985835 IC50 = 1800 nM T02506 CG8O2K 145986244 IC50 = 96 nM T02506 CN91YC 145986320 EC50 = 158 nM T02506 CF49OP 145986577 IC50 = 4677 nM T02506 CMQK52 145986591 IC50 = 23 nM T02506 C28LAH 145986759 IC50 = 769 nM T02506 CA1D2B 145987043 IC50 = 48 nM T02506 CPRH38 145987084 EC50 = 1003 nM T02506 CF9S0O 145987265 IC50 = 407 nM T02506 CKYW98 145988223 EC50 = 204 nM T02506 CK5RV0 145988666 EC50 > 10000 nM T02506 C09MNB 145988825 IC50 = 67 nM T02506 CW0C8Y 145989462 EC50 = 1831 nM T02506 CX74YQ 145989561 EC50 = 199 nM T02506 CSF03L 145989681 IC50 = 41 nM T02506 CR0LK9 145989755 EC50 = 721 nM T02506 COI2R8 145991129 EC50 = 219 nM T02506 C2NH3M 145991296 IC50 = 413 nM T02506 CP4V8N 145991796 IC50 = 179 nM T02506 CQ1WY2 146183836 IC50 = 0.79 nM T02506 C04KLS 146428237 IC50 = 0.24 nM T02506 C9K2RG 146428250 IC50 = 0.61 nM T02506 CWG2N1 146567341 IC50 = 0.7 nM T02506 CFNR34 146567342 IC50 = 0.49 nM T02506 C43PZX 146567347 IC50 = 0.37 nM T02506 C8ZL7B 146567366 IC50 = 0.82 nM T02506 CFD3E8 146567377 IC50 = 0.5 nM T02506 C5G2BR 146567380 IC50 = 0.3 nM T02506 C3C1XK 146567381 IC50 = 0.7 nM T02506 C46GUI 149822983 IC50 = 0.5 nM T02506 C6Y8BH 155510359 IC50 = 2980 nM T02506 CF8PO7 155511409 IC50 = 2.4 nM T02506 CCGY16 155511936 IC50 = 0.3162 nM T02506 C7VS5G 155511937 IC50 = 1240 nM T02506 CIJ4K9 155512714 IC50 = 27 nM T02506 CVCK17 155513135 IC50 > 10000 nM T02506 C2PU1J 155513315 IC50 = 1700 nM T02506 CGKQ42 155513962 IC50 = 0.021 nM T02506 CMQC26 155515404 IC50 = 1658 nM T02506 CP1L3J 155516697 IC50 > 10000 nM T02506 CL80FT 155516984 EC50 = 2 nM T02506 CFJO71 155518954 IC50 = 0.17 nM T02506 CLR23U 155519218 IC50 > 5000 nM T02506 CY94AM 155520303 IC50 = 90 nM T02506 C5CXT0 155520789 EC50 = 20 nM T02506 CMWI40 155521404 IC50 = 1780 nM T02506 C7LVS8 155521699 IC50 = 0.8 nM T02506 C4RK1P 155522067 IC50 = 15 nM T02506 C3LNK9 155522178 IC50 = 63.1 nM T02506 CSE31P 155522268 IC50 = 0.28 nM T02506 C9MAF1 155525071 IC50 = 0.42 nM T02506 C4PIM5 155526909 IC50 = 7.5 nM T02506 CAJW03 155527870 IC50 = 5.7 nM T02506 CSLJ15 155528850 IC50 > 10000 nM T02506 C0GY8X 155529068 IC50 = 0.7943 nM T02506 CUO74Y 155529729 EC50 = 0.6 nM T02506 CH42RB 155530321 IC50 = 0.07 nM T02506 CE4S3C 155533437 IC50 = 4.71 nM T02506 C0TW8H 155534195 IC50 = 94 nM T02506 CC5HJ6 155535796 IC50 > 10000 nM T02506 CI5T9E 155536687 EC50 = 1.3 nM T02506 CS06LK 155537645 EC50 = 140 nM T02506 CYS47I 155537918 IC50 > 100 nM T02506 C9EW1F 155538055 IC50 = 0.2 nM T02506 CH3V8J 155538711 EC50 = 427 nM T02506 CB3CY8 155538987 IC50 = 2500 nM T02506 COP7X8 155539171 IC50 > 10000 nM T02506 C4ID8Q 155539669 IC50 > 5000 nM T02506 CA2G8E 155539747 IC50 = 0.3162 nM T02506 C90XVB 155539810 IC50 = 25.12 nM T02506 CKF67H 155540121 IC50 = 1.995 nM T02506 C2RAP5 155540472 IC50 > 100 nM T02506 CMT91D 155540730 IC50 = 2300 nM T02506 C31CNR 155541121 IC50 > 5000 nM T02506 C8MPH9 155541236 IC50 = 1.259 nM T02506 CL53BE 155543769 IC50 = 2460 nM T02506 CU9A7M 155544127 Ki = 25 nM T02506 CF6TH5 155546055 IC50 = 2.5 nM T02506 CT0ON6 155546145 IC50 = 31 nM T02506 CP9Y8J 155548583 IC50 > 5000 nM T02506 C2PUT5 155549053 EC50 = 93 nM T02506 CA5G2T 155551013 IC50 > 10000 nM T02506 CRS02E 155551888 IC50 = 2330 nM T02506 CS9D3O 155552434 IC50 > 100 nM T02506 CF68WS 155552480 IC50 = 100 nM T02506 C5MHU4 155552943 IC50 > 5000 nM T02506 C1DC4A 155553793 IC50 = 30 nM T02506 C5S9LI 155556292 IC50 > 10000 nM T02506 CT3F5K 155556316 IC50 = 0.5 nM T02506 CY1S3T 155557113 IC50 = 8.15 nM T02506 C7AJZ5 155559268 IC50 = 1142 nM T02506 CHI07R 155559518 EC50 = 1 nM T02506 CLJ4A1 155559849 IC50 > 100 nM T02506 C2D6ZM 155561414 EC50 > 500 nM T02506 CV5I6E 155562017 IC50 = 37 nM T02506 C4CJ7W 155562234 IC50 = 250000 nM T02506 C9KY5I 155562382 IC50 > 10000 nM T02506 CSJQ98 155562658 IC50 = 22.67 nM T02506 C5NR7H 155562810 IC50 = 213 nM T02506 C48NOU 155563946 EC50 = 0.2 nM T02506 C7JMZ0 155564173 IC50 = 0.3 nM T02506 CQ97FI 155564996 IC50 = 72 nM T02506 CWK95R 155565459 IC50 > 10000 nM T02506 CY71WP 155565677 IC50 > 10000 nM T02506 C2UTY4 155566549 IC50 = 0.631 nM T02506 CT7OB2 155566794 IC50 = 19.95 nM T02506 C4C9PF 155566802 IC50 = 0.3162 nM T02506 C4HFX0 155566914 EC50 = 193 nM T02506 CMX67L 155567147 IC50 = 2116 nM T02506 C2NBO7 155567224 IC50 = 0.3 nM T02506 CY28HU 155567231 IC50 > 5000 nM T02506 C76EWQ 155567785 IC50 = 1.76 nM T02506 C4ZQ7D 155568522 IC50 = 1 nM T02506 CJRS26 155568547 IC50 = 6300 nM T02506 C4JTH2 155568868 IC50 > 5000 nM T02506 C5I0QV 155569431 IC50 = 0.08 nM T02506 CVD17E 10087534 EC50 = 380 nM T02506 C0RGJ9 44389594 EC50 = 1.1 nM T02506 D00CWN 135987619 Ki = 310 nM T02506 D00DJX 44597742 IC50 = 11 nM T02506 D00HZT 135449109 IC50 = 780 nM T02506 D00IXB 10445833 IC50 = 101 nM T02506 D00NEK 44405867 IC50 = 8310 nM T02506 D00RIX 5280443 IC50 = 1253 nM T02506 D00URP 10399473 IC50 = 1030 nM T02506 D00XLU 44407802 EC50 = 242 nM T02506 D00ZBL 135458122 IC50 = 727 nM T02506 D01AHL 44412953 IC50 > 10000 nM T02506 D01CYI 11579721 IC50 = 53640 nM T02506 D01GPY 10192794 IC50 = 40 nM T02506 D01IAT 10171410 IC50 = 2642 nM T02506 D01KJU 6102690 IC50 = 91 nM T02506 D01KSR 135495079 IC50 = 2765 nM T02506 D01QXL 9993627 IC50 = 153 nM T02506 D01SWO 9901869 IC50 = 35 nM T02506 D01TUB 135519319 IC50 = 213 nM T02506 D01WCA 656936 IC50 = 176 nM T02506 D01XCA 44407801 EC50 = 534 nM T02506 D02DML 5281707 IC50 = 11 nM T02506 D02EJM 136048731 IC50 = 775 nM T02506 D02GLM 9994500 Ki = 2800 nM T02506 D02HGS 135502634 IC50 = 632 nM T02506 D02JJU 135492380 IC50 = 3800 nM T02506 D02LCC 135442595 IC50 = 1200 nM T02506 D02OKF 10308197 IC50 = 10 nM T02506 D02RQP 6623 EC50 = 290 nM T02506 D02TPO 10323679 IC50 = 10 nM T02506 D02WRU 11201035 Ki = 2222 nM T02506 D02WSA 11579722 IC50 = 75588 nM T02506 D02XVV 10399376 IC50 > 10000 nM T02506 D02ZSX 61253 IC50 = 8740 nM T02506 D03BOO 25128804 Ki = 4100 nM T02506 D03CBX 135454802 IC50 = 212 nM T02506 D03DVM 10131379 IC50 = 31 nM T02506 D03GYS 135499774 IC50 = 498 nM T02506 D03NTD 9878556 Ki = 132 nM T02506 D03QHG 16066665 IC50 = 216 nM T02506 D03RYU 135522275 IC50 = 82 nM T02506 D03XEU 10286022 IC50 = 483 nM T02506 D04EAY 135474202 IC50 = 3000 nM T02506 D04SAO 9799518 EC50 = 1.7 nM T02506 D04TPC 25130896 Ki > 7300 nM T02506 D04WHH 135519317 IC50 = 390 nM T02506 D05EOW 102614 EC50 = 3.4 nM T02506 D05FUY 10149584 IC50 = 43 nM T02506 D05JKC 135546593 IC50 = 464 nM T02506 D05JPW 135409725 IC50 = 2557 nM T02506 D05KXP 44418726 IC50 = 1017 nM T02506 D05LQD 10082995 IC50 > 10000 nM T02506 D05PNP 11064571 IC50 = 26200 nM T02506 D05YIU 10236250 IC50 = 6.8 nM T02506 D06DDT 5315502 EC50 = 1590 nM T02506 D06OAL 135442585 IC50 = 537 nM T02506 D06SCS 135418373 IC50 = 155 nM T02506 D07HBQ 25128814 IC50 = 2400 nM T02506 D07LUI 11459006 IC50 = 211 nM T02506 D07TGS 3017674 IC50 = 150 nM T02506 D07TGW 135857091 IC50 = 20 nM T02506 D07VPM 135409756 IC50 = 1300 nM T02506 D07XBD 10308075 IC50 = 282 nM T02506 D07XUY 44418717 IC50 = 5245 nM T02506 D08FLV 135474625 IC50 = 819 nM T02506 D08GWS 46919124 Ki = 25.43 nM T02506 D08HCF 135496133 IC50 = 5000 nM T02506 D08LVT 44407806 IC50 = 1371 nM T02506 D08SJL 135524856 IC50 = 1500 nM T02506 D08VDX 10214699 IC50 = 30 nM T02506 D08WDN 135496123 IC50 = 6100 nM T02506 D09CQC 135471161 IC50 = 902 nM T02506 D09DEK 10171409 IC50 = 442 nM T02506 D09FWP 11368353 IC50 > 5000 nM T02506 D09FWS 135430317 IC50 = 634 nM T02506 D09NFD 6852176 IC50 = 320 nM T02506 D09NOH 44418728 IC50 = 140 nM T02506 D09PXU 9991961 IC50 = 4610 nM T02506 D09TQE 135528620 IC50 = 1570 nM T02506 D09ULU 2368773 IC50 = 404 nM T02506 D09UQU 10029432 IC50 = 64 nM T02506 D09UWI 14905189 EC50 = 2350 nM T02506 D09WEK 135503667 EC50 = 390 nM T02506 D0AD3U 135528621 IC50 = 8430 nM T02506 D0AD8G 44407887 IC50 = 235 nM T02506 D0AU0M 637542 EC50 = 16120 nM T02506 D0B1HP 135526958 IC50 = 815 nM T02506 D0C4VX 135407148 IC50 = 52 nM T02506 D0C5FY 10331951 IC50 = 654 nM T02506 D0C6AP 10285954 IC50 = 114 nM T02506 D0C6UR 49863610 Ki = 13.66 nM T02506 D0C9XK 135545334 IC50 = 2410 nM T02506 D0C9XW 11276767 IC50 = 13000 nM T02506 D0CC6R 10125290 IC50 = 24 nM T02506 D0D1LB 44418733 IC50 = 503 nM T02506 D0DK9S 135454786 IC50 = 6240 nM T02506 D0F1SS 44605900 EC50 > 10000 nM T02506 D0F8LS 135524867 IC50 = 18 nM T02506 D0FD6Z 10308090 IC50 = 22 nM T02506 D0H1CO 10244394 IC50 = 1880 nM T02506 D0H2FI 10308268 IC50 = 709 nM T02506 D0H5HI 9993278 IC50 = 468 nM T02506 D0H6MZ 25133613 IC50 = 7300 nM T02506 D0H8PI 10308021 IC50 = 22 nM T02506 D0H8ZT 135525228 IC50 = 37 nM T02506 D0HD2G 4788 IC50 = 300 nM T02506 D0HM8Y 44408971 IC50 = 1170 nM T02506 D0HR8L 11447703 IC50 = 1452 nM T02506 D0I1NX 10246180 EC50 = 0.15 nM T02506 D0I5HZ 44405888 IC50 = 1800 nM T02506 D0I5VJ 135520257 IC50 = 55883 nM T02506 D0J0AG 135421237 IC50 = 1140 nM T02506 D0J2NG 44418724 IC50 = 392 nM T02506 D0J3PM 44407886 EC50 = 1985 nM T02506 D0J6KN 135511848 IC50 = 40 nM T02506 D0K0IC 13896065 IC50 = 24 nM T02506 D0K0TR 11356877 IC50 1000000 nM T02506 D0K1TW 135443280 IC50 = 5280 nM T02506 D0K5LX 135566322 IC50 = 48 nM T02506 D0K6TE 10286087 IC50 = 107 nM T02506 D0K7HR 135409729 IC50 = 504 nM T02506 D0K8QD 63059 EC50 = 0.015 nM T02506 D0L0RK 44407885 EC50 = 1430 nM T02506 D0L2MU 10286352 IC50 = 1.5 nM T02506 D0L3AX 236868 IC50 = 638 nM T02506 D0L6IQ 135424609 IC50 = 6630 nM T02506 D0LI0M 44418723 IC50 = 383 nM T02506 D0M0RS 11560224 Ki > 1000 nM T02506 D0M0XL 11414445 IC50 = 884 nM T02506 D0M4LQ 44407804 EC50 = 705 nM T02506 D0MY8V 10308207 IC50 = 92 nM T02506 D0N0OY 135405741 IC50 = 1227 nM T02506 D0NN0V 637048 IC50 = 10200 nM T02506 D0O2KP 12133211 IC50 = 58 nM T02506 D0O5KR 10060956 IC50 = 335 nM T02506 D0O6FX 10061675 IC50 = 237 nM T02506 D0O9NE 5388063 Ki = 261 nM T02506 D0OV3S 11782482 IC50 = 50 nM T02506 D0P4SR 11716633 EC50 = 17 nM T02506 D0P6FN 10125342 IC50 = 174 nM T02506 D0P7PK 77020 IC50 = 6950 nM T02506 D0P8PK 10192730 IC50 = 230 nM T02506 D0Q4VG 135458016 IC50 = 25 nM T02506 D0Q6MS 11141183 IC50 = 30 nM T02506 D0R7AG 135486039 IC50 = 190 nM T02506 D0R7QY 127676 EC50 = 2600 nM T02506 D0S0SZ 135409723 IC50 = 481 nM T02506 D0S2ZJ 135430305 IC50 = 2353 nM T02506 D0S5RI 11547961 Ki = 13.01 nM T02506 D0S6NV 10149684 IC50 = 266 nM T02506 D0S8AV 509245 IC50 = 57 nM T02506 D0S8EB 11777167 IC50 = 1210 nM T02506 D0SR8Q 11458674 IC50 = 3405 nM T02506 D0SY2M 5281708 IC50 = 450 nM T02506 D0U0ZE 44408769 IC50 = 585 nM T02506 D0U2VA 4369550 IC50 = 117 nM T02506 D0U7KV 201385 IC50 = 94.8 nM T02506 D0UV9G 10125182 IC50 = 1345 nM T02506 D0V6KJ 10214708 IC50 = 10.3 nM T02506 D0V7OK 6366969 IC50 = 7 nM T02506 D0V7QZ 135528624 IC50 = 139 nM T02506 D0V7ZI 135476471 EC50 = 98 nM T02506 D0VN2R 10171886 IC50 = 1231 nM T02506 D0W0LG 44418722 IC50 = 155 nM T02506 D0W2YR 135522274 IC50 = 5110 nM T02506 D0W3FF 135503567 IC50 = 1900 nM T02506 D0W4WF 100801 IC50 = 240 nM T02506 D0W5HT 44418725 IC50 = 436 nM T02506 D0WM5O 5322399 Ki > 10000 nM T02506 D0WP6A 5348729 IC50 > 10000 nM T02506 D0X0RJ 9848809 IC50 = 76 nM T02506 D0X2VK 9945207 IC50 = 4.3 nM T02506 D0X4VN 10236221 IC50 = 92 nM T02506 D0X6LK 10823890 IC50 = 2700 nM T02506 D0X7DJ 10308206 IC50 = 27 nM T02506 D0X7SR 10246505 EC50 = 50 nM T02506 D0XC3V 10871661 IC50 = 500 nM T02506 D0XF9F 135484659 Ki = 2.7 nM T02506 D0XS0R 44433505 Ki > 1100 nM T02506 D0Y2LJ 44418729 IC50 = 80 nM T02506 D0Y4NJ 11784736 IC50 = 0.28 nM T02506 D0Y8UF 5040063 EC50 = 0.1 nM T02506 D0Y9BO 135461982 IC50 = 93 nM T02506 D0YH4T 10062042 IC50 = 35 nM T02506 D0YW4C 135494488 IC50 = 447 nM T02506 D0Z0UC 11638264 EC50 = 7 nM T02506 D0Z9ZY 23582387 EC50 = 1543 nM T02506 D0ZT4U 10214633 IC50 = 77 nM T92328 CS3PR5 5114 Ki = 1.8 nM T92328 C0CYV1 6413514 EC50 > 100000 nM T92328 C5CXD3 10328662 EC50 = 14700 nM T92328 C58IAT 11845229 IC50 = 6000 nM T92328 C56OCS 11845762 EC50 = 11000 nM T70309 D08IWD 57363 IC50 = 19.8 ug.mL-1 T70309 D0A9YA 6918296 IC50 = 4 nM T70309 D02KRI 68741 Ki = 410 nM T70309 D0J3CT 178077 IC50 = 3 nM T70309 D0P9EL 10220187 Ki = 5.8 nM T70309 D0Z9UB 166562 IC50 = 2.3 nM T70309 C3EP4O 81146 Ki > 2500 nM T70309 CE7GN4 116469 Ki = 315 nM T70309 CMXV58 130227 Ki = 1600 nM T70309 CSD84A 132992 IC50 = 16 nM T70309 CBY29G 260801 Ki = 460 nM T70309 C6SDC5 322615 IC50 = 6500 nM T70309 CTX0Z3 327169 IC50 > 20 ug.mL-1 T70309 CT41AK 348591 Ki > 2500 nM T70309 CG21HL 849844 IC50 > 4 ug.mL-1 T70309 C20JCF 2735497 Ki > 2500 nM T70309 CJ9LZ7 3051101 IC50 > 20 ug.mL-1 T70309 C4QJ7Z 4777878 Ki > 2500 nM T70309 C2URF8 5290170 IC50 = 0.2 ug.mL-1 T70309 CU4NO6 9798052 IC50 = 79.43 nM T70309 CVF6K7 9805325 IC50 = 40 nM T70309 C6VPY0 9859767 IC50 = 7.943 nM T70309 C8G3MQ 9860236 Ki = 120 nM T70309 C68XWT 9881419 IC50 = 1800 nM T70309 CRO5V7 9882015 Ki = 1200 nM T70309 C87KNG 9914880 IC50 = 2.4 nM T70309 CN0TU8 9915286 IC50 = 50 nM T70309 C3LF1G 9915313 IC50 = 20 nM T70309 CA3DS4 9981612 IC50 = 1.77 nM T70309 C3ZP7E 9981699 IC50 = 5.6 nM T70309 COM8P4 9991591 IC50 = 35 nM T70309 C7BWP9 10006358 IC50 = 310 nM T70309 CY0KZ4 10022795 IC50 = 3.4 nM T70309 CQA6M3 10040787 IC50 = 0.15 ug.mL-1 T70309 CJC2B8 10049013 IC50 = 8.1 nM T70309 CCP81A 10059992 IC50 = 60 nM T70309 C7LY9P 10064026 Ki = 500 nM T70309 CUJ3V9 10064949 IC50 = 152 nM T70309 C1R9SW 10076629 IC50 = 130 nM T70309 C2MRU3 10082004 IC50 = 560 nM T70309 CLDT58 10083173 IC50 = 0.2 ug.mL-1 T70309 CEZG10 10105225 IC50 = 11 nM T70309 CMGW89 10105927 IC50 = 120 nM T70309 C2J3SN 10130763 IC50 = 32.36 nM T70309 CH4UD5 10220542 Ki = 2.7 nM T70309 C9IS3Z 10243712 Ki = 17 nM T70309 C3FGC8 10254719 IC50 = 574 nM T70309 C2AK6N 10264096 Ki = 15 nM T70309 C7RH6M 10266307 IC50 = 8.1 nM T70309 CR9BY2 10318958 IC50 = 0.91 nM T70309 C2DW4G 10330957 IC50 = 3200 nM T70309 CX9CU2 10331550 IC50 = 320 nM T70309 CV93KQ 10355313 IC50 = 120 nM T70309 C8KG1C 10363135 IC50 = 20 nM T70309 CVM5I4 10365419 IC50 = 9.57 nM T70309 CGVX26 10376044 IC50 = 10000 nM T70309 CO9ST8 10377317 IC50 = 14.4 nM T70309 CIRV78 10380223 Ki = 26 nM T70309 CO4XP8 10386420 IC50 = 2.19 nM T70309 C3L5QA 10387222 IC50 = 7.25 nM T70309 C2HVN8 10411536 Ki = 6.9 nM T70309 CJV3F4 10413543 IC50 = 25 nM T70309 CQY7J1 10422666 Ki = 320 nM T70309 CO8U9D 10436202 IC50 = 62 nM T70309 C12INV 10445491 Ki = 20 nM T70309 C42TKU 10453975 IC50 > 1000 nM T70309 CNL09S 10466539 IC50 = 460 nM T70309 C5TDF3 10467173 IC50 = 3600 nM T70309 C1TM7R 10469538 IC50 = 107 nM T70309 C5N7PW 10500864 IC50 = 410 nM T70309 CGF70C 10513499 IC50 = 5310 nM T70309 C5HQ4N 10514266 IC50 = 15.8 nM T70309 COB59J 10514668 IC50 = 204 nM T70309 C51MLZ 10540212 IC50 = 299 nM T70309 C2FHE3 10586600 IC50 = 188 nM T70309 CWL9M1 10587522 IC50 = 8.5 nM T70309 CT3BX5 10588455 IC50 = 409 nM T70309 C80SRG 10656221 IC50 = 376 nM T70309 C10EJO 10656222 IC50 = 185 nM T70309 CVSW93 10658050 IC50 = 1880 nM T70309 C3Q8MZ 10681970 IC50 = 9100 nM T70309 CIV2R1 10682868 IC50 = 15.6 nM T70309 CM72CD 10727316 IC50 = 176 nM T70309 CY6D7I 10737132 IC50 = 1134 nM T70309 CNY1R4 10823556 IC50 = 459 nM T70309 C1J6UG 10847272 IC50 = 49 nM T70309 C6QJ5E 10848122 IC50 = 5310 nM T70309 CM28KN 10850018 IC50 > 100000 nM T70309 CIS0Y3 10873561 IC50 = 700 nM T70309 C9SUP2 10971743 IC50 = 1300 nM T70309 CL32RH 11122765 IC50 = 75 nM T70309 CT1WB4 11160874 IC50 = 178 nM T70309 CZ3YU8 11161937 IC50 = 218.78 nM T70309 C5LX1F 11163404 IC50 = 942 nM T70309 C1Z0SH 11172491 IC50 = 21.38 nM T70309 CPY7N1 11173292 IC50 = 117 nM T70309 C3XTI0 11185533 IC50 = 79 nM T70309 CAR5P2 11220790 IC50 = 14.13 nM T70309 C7WV2R 11229432 IC50 = 8400 nM T70309 CO0RP5 11243912 IC50 = 1000 nM T70309 CDIA87 11244952 IC50 = 1047.13 nM T70309 C04TKS 11268166 IC50 = 93 nM T70309 CX73IS 11300738 IC50 = 128 nM T70309 CRZ4X7 11301454 IC50 = 8.71 nM T70309 CO1LZ4 11302657 IC50 = 194 nM T70309 C0SHF3 11303884 IC50 = 954.99 nM T70309 CL90FN 11313212 IC50 = 111 nM T70309 CQ5H0U 11315272 IC50 = 560 nM T70309 CU1CX8 11363043 IC50 = 389.05 nM T70309 CE0V6Q 11381020 IC50 = 724.44 nM T70309 C4FB8M 11382643 IC50 = 92.9 nM T70309 C7ZYN4 11382644 IC50 = 93 nM T70309 CV1Z2R 11429133 IC50 = 83.7 nM T70309 C56TXQ 11442425 IC50 = 147.91 nM T70309 CRHX97 11472526 IC50 = 380.19 nM T70309 CA6UH4 11482868 IC50 = 131.83 nM T70309 C9SXK5 11483152 IC50 = 169.82 nM T70309 C31TGA 11486129 IC50 = 120.23 nM T70309 CI8RC4 11723581 IC50 = 620 nM T70309 C0FJS4 11736622 IC50 = 14.13 nM T70309 C2JE6U 11746372 IC50 > 20 ug.mL-1 T70309 CR5N7I 11755506 IC50 = 0.9 nM T70309 CGU4O8 11772392 IC50 = 97.72 nM T70309 CH8CU1 11820650 IC50 = 600 nM T70309 C5DO4L 11820651 IC50 = 2300 nM T70309 C96DPL 11855879 IC50 = 770 nM T70309 CW4I5R 12012173 IC50 = 377 nM T70309 CM9DS4 12012174 IC50 = 183 nM T70309 CLQ19M 12969972 IC50 = 4300 nM T70309 C8EW5G 15337643 IC50 = 34.67 nM T70309 C7LX0N 15506062 IC50 = 1300 nM T70309 CR16DG 18542500 IC50 = 312 nM T70309 CRD8P6 18542503 IC50 = 141 nM T70309 C0NMF9 18654192 IC50 = 120 nM T70309 C5AN0E 19707315 IC50 = 1000 nM T70309 CMH8W6 19707318 IC50 = 34.67 nM T70309 CGM4S5 19707325 IC50 = 114.82 nM T70309 CANJ35 19707345 IC50 = 562.34 nM T70309 CSA2C6 19707363 IC50 = 32.36 nM T70309 C0T4DC 19707381 IC50 = 114.82 nM T70309 CF9H2E 19791557 IC50 = 1000 nM T70309 CCOE86 19791558 IC50 = 151.36 nM T70309 C9V5RQ 19927034 Ki = 1200 nM T70309 CV0JP1 22909503 IC50 = 60.26 nM T70309 C0R3DQ 22909504 IC50 = 89.13 nM T70309 C2DQO8 24180522 IC50 = 840 nM T70309 CU6HP4 44264624 IC50 = 10.5 nM T70309 C9C4RK 44271130 IC50 = 3.22 nM T70309 CSV64F 44271133 IC50 = 2.42 nM T70309 C4MD0O 44271147 IC50 = 3700 nM T70309 CCO08D 44271150 IC50 = 3.31 nM T70309 CKYH52 44271172 IC50 = 10.6 nM T70309 C4AWP7 44271177 IC50 = 7.31 nM T70309 CIZ64F 44271186 IC50 = 9.53 nM T70309 C7MI6C 44271188 IC50 = 2.35 nM T70309 CT4XU9 44271189 IC50 > 100 nM T70309 C6R0WD 44271195 IC50 = 16.9 nM T70309 C3JD5Z 44271203 IC50 = 5.08 nM T70309 CD1E0B 44271224 IC50 = 29 nM T70309 C2NSM8 44271225 IC50 = 4.56 nM T70309 C1FQ6O 44271232 IC50 = 11.8 nM T70309 C8YEA5 44271245 IC50 = 1900 nM T70309 C45ZCB 44271246 IC50 > 100 nM T70309 CE17GD 44271251 IC50 = 5.63 nM T70309 C0W1DK 44271252 IC50 = 11.9 nM T70309 C1D3AE 44271258 IC50 = 2.11 nM T70309 C2VY7C 44271268 IC50 = 3.05 nM T70309 C2NWJ0 44271274 IC50 = 2.93 nM T70309 CM02PT 44271279 IC50 = 11.2 nM T70309 CU3P4D 44271283 IC50 = 59.8 nM T70309 C7D2RT 44271314 IC50 = 32.8 nM T70309 CBA70P 44271320 IC50 = 5.44 nM T70309 CWI8M6 44274870 IC50 = 14 nM T70309 CX6BV1 44274932 IC50 = 5.6 nM T70309 C8HK3W 44274947 IC50 > 1000 nM T70309 CSN05C 44275112 IC50 = 8 nM T70309 CWP7D4 44275145 IC50 = 0.5 nM T70309 CB7R1A 44275146 IC50 = 1.7 nM T70309 CGJ7T9 44275147 IC50 = 19.1 nM T70309 C8CI9L 44275160 Ki = 9 nM T70309 CWXD82 44275204 IC50 = 8.1 nM T70309 C7HV2D 44275216 IC50 = 981 nM T70309 CASH41 44275218 IC50 = 120.2 nM T70309 C73HPZ 44275234 IC50 = 350 nM T70309 CC6U2N 44275245 IC50 = 20 nM T70309 CQR65M 44275322 IC50 = 134 nM T70309 C0DQM8 44275323 IC50 = 3.3 nM T70309 C15CZH 44275436 IC50 = 10 nM T70309 CV0LC3 44277746 Ki = 4000 nM T70309 C5KH4A 44287925 IC50 = 2100000 nM T70309 CY2IC1 44287935 IC50 = 3200000 nM T70309 CH2ZT5 44288066 IC50 = 2780000 nM T70309 CB5VS4 44299604 IC50 = 1450 nM T70309 CK2RJ9 44299652 IC50 = 23 nM T70309 CCED35 44314879 Ki = 4900 nM T70309 C3TK6L 44314902 Ki = 1900 nM T70309 C2AC1R 44314907 Ki = 1900 nM T70309 CGI6N3 44314943 Ki = 1900 nM T70309 CLM49Y 44315410 Ki = 6.4 nM T70309 CF7R9X 44315430 Ki = 48 nM T70309 CJM7E9 44315474 Ki = 8.5 nM T70309 CN58ZU 44315547 Ki = 340 nM T70309 CTP9N0 44315618 Ki = 82 nM T70309 C2DKW4 44315657 Ki = 5900 nM T70309 CI3E5Z 44315682 Ki = 6.2 nM T70309 CO7ZU0 44315685 Ki = 280 nM T70309 C9A0YC 44315700 Ki = 8.6 nM T70309 C2UC3Q 44315719 IC50 > 20 ug.mL-1 T70309 CVD24Q 44315722 Ki = 40000 nM T70309 CGO49I 44315724 IC50 > 4 ug.mL-1 T70309 C2NGO7 44315730 IC50 = 13.6 ug.mL-1 T70309 C5Z9SV 44315735 IC50 > 20 ug.mL-1 T70309 CVAG48 44315739 Ki = 1400 nM T70309 CGXN06 44315740 Ki = 87 nM T70309 CB6I7M 44315750 IC50 > 4 ug.mL-1 T70309 C05YTO 44315755 Ki = 1300 nM T70309 CP49RD 44315756 Ki = 7800 nM T70309 CT0QB5 44315757 Ki = 3400 nM T70309 CZHB84 44315759 Ki = 5800 nM T70309 CM0KD2 44315819 Ki = 3.1 nM T70309 CVYR32 44315864 Ki = 74 nM T70309 C0DA9R 44315908 Ki = 60 nM T70309 CV3X6A 44315969 Ki = 24000 nM T70309 C1WG6H 44315970 Ki = 10000 nM T70309 C2ORG3 44315992 Ki = 10000 nM T70309 CD27VS 44316012 Ki = 10000 nM T70309 C9XR5K 44316040 Ki = 8300 nM T70309 C5C3VS 44316042 Ki = 280 nM T70309 C8SKX0 44316063 Ki = 2400 nM T70309 C4UR6E 44316076 Ki = 1300 nM T70309 C2NG1P 44316077 Ki = 180 nM T70309 C7NOY4 44322148 Ki = 0.13 nM T70309 CJ4P8B 44322225 IC50 = 60 nM T70309 CXBF03 44329329 IC50 = 127 nM T70309 CJGD39 44338101 IC50 = 19 nM T70309 CM85RX 44338102 IC50 = 11 nM T70309 C6M9QA 44338152 IC50 = 12.5 nM T70309 C4IKG5 44338162 IC50 = 20.5 nM T70309 C3XU2H 44338163 IC50 = 6.8 nM T70309 C2V5CD 44338164 IC50 = 18.2 nM T70309 C4B0RA 44338187 IC50 = 22.5 nM T70309 C6T0PA 44338193 IC50 = 20.9 nM T70309 CBXO72 44338225 IC50 = 94 nM T70309 C9TSK2 44338226 IC50 = 28.7 nM T70309 CVD4I2 44338231 IC50 = 14.5 nM T70309 CIF8K9 44338238 IC50 = 595 nM T70309 C8REO3 44338254 IC50 = 23 nM T70309 CX9EB7 44338255 IC50 = 7.9 nM T70309 C1D9TE 44338287 IC50 > 1000 nM T70309 CYMP02 44338289 IC50 = 19 nM T70309 CIQ50X 44338290 IC50 = 12.9 nM T70309 CQX4H3 44338298 IC50 = 154 nM T70309 C4ZTP0 44338299 IC50 = 130 nM T70309 CWY72O 44338303 IC50 = 34.9 nM T70309 CY87ER 44338307 IC50 = 14 nM T70309 C79VZY 44338311 Ki = 4200 nM T70309 CQJ8F7 44338320 IC50 = 38.3 nM T70309 CFC71N 44338329 IC50 = 14 nM T70309 CD20EX 44338333 IC50 = 26 nM T70309 CO5ME9 44338343 IC50 = 614 nM T70309 CQM89S 44338379 IC50 = 350 nM T70309 CG4CX1 44338395 IC50 = 17.2 nM T70309 C3HTB0 44338396 IC50 = 24.6 nM T70309 C8Y1SR 44338430 IC50 = 30.3 nM T70309 C03SKL 44338440 IC50 = 5.8 nM T70309 CS84KM 44338457 IC50 = 52 nM T70309 C6G3QX 44338558 IC50 = 120.2 nM T70309 C53AIN 44338631 IC50 = 17.2 nM T70309 C56QUC 44338632 IC50 = 74 nM T70309 C3WMT4 44338668 IC50 = 12 nM T70309 CULP10 44338682 IC50 = 120 nM T70309 CGA5E4 44343784 IC50 = 188 nM T70309 CO0XF3 44345135 IC50 = 459 nM T70309 C17TJS 44345150 IC50 = 346 nM T70309 CDQC58 44345345 IC50 = 14.4 nM T70309 CY5QP4 44348908 IC50 = 137 nM T70309 CK9QZ1 44348923 IC50 = 9100 nM T70309 C8U2DT 44348944 IC50 = 2700 nM T70309 CWPS98 44349957 IC50 = 8.4 nM T70309 C9ECO7 44349958 IC50 = 9.5 nM T70309 CPVY25 44349965 IC50 = 4.3 nM T70309 C4WNL3 44350041 IC50 = 1.7 nM T70309 CMN9R2 44350093 IC50 = 0.6 nM T70309 CSO78L 44350227 IC50 = 134 nM T70309 CCO46E 44350228 IC50 = 5.7 nM T70309 C4YR2P 44350229 IC50 = 42 nM T70309 C0E8OQ 44350239 IC50 = 20 nM T70309 C3FV2X 44350245 IC50 = 5 nM T70309 CR6LZ1 44350246 IC50 > 1000 nM T70309 C1RHZ6 44350258 IC50 = 2 nM T70309 C2SRP4 44350270 IC50 = 2.7 nM T70309 C0A6MU 44350284 IC50 = 3.3 nM T70309 CDA84X 44350285 IC50 = 1.6 nM T70309 C0BV4E 44350286 IC50 > 1000 nM T70309 CE90TU 44350289 IC50 = 2.6 nM T70309 CMA2Z5 44350291 IC50 = 58 nM T70309 C97TQC 44350292 IC50 = 2.5 nM T70309 CCE5U6 44350293 IC50 = 8.6 nM T70309 C7N9MR 44350326 IC50 = 2.6 nM T70309 CT1SC9 44350327 IC50 = 9.5 nM T70309 CHQ9T5 44350334 IC50 > 1000 nM T70309 CI7S0L 44350481 IC50 = 19.1 nM T70309 C3G7LK 44351555 IC50 > 10000 nM T70309 CH9XO4 44351556 IC50 = 63 nM T70309 C7S8HU 44351573 IC50 = 32 nM T70309 C5GSO0 44351575 IC50 > 10000 nM T70309 CR83SY 44351601 IC50 > 10000 nM T70309 C9UA2Q 44351707 IC50 = 6 nM T70309 CTS3J6 44351715 IC50 > 10000 nM T70309 CGMQ98 44351716 IC50 = 59 nM T70309 C7C5WX 44351747 IC50 > 10000 nM T70309 CA8M1B 44351848 IC50 = 21 nM T70309 CJM80V 44358932 IC50 = 1600 nM T70309 CSN53U 44363198 Ki > 2500 nM T70309 C7U5PF 44391584 IC50 = 268 nM T70309 CLF8E2 44391595 IC50 = 463 nM T70309 COAB23 44391699 IC50 = 160 nM T70309 C9VUS0 44391700 IC50 = 138 nM T70309 CM4H1G 44391702 IC50 = 361 nM T70309 CK34ES 44391712 IC50 = 149 nM T70309 C52WFS 44391720 IC50 = 225 nM T70309 CB69UH 44391721 IC50 = 271 nM T70309 C18RXO 44391730 IC50 = 1000 nM T70309 CIC71T 44391731 IC50 = 42 nM T70309 CV40UR 44391732 IC50 = 272 nM T70309 C79CYJ 44391758 IC50 = 116 nM T70309 CZ7Q6H 44391760 IC50 = 707 nM T70309 CY4PH3 44391764 IC50 = 209 nM T70309 C6TM0S 44391773 IC50 = 1400 nM T70309 CBZ56Q 44391891 IC50 = 6990 nM T70309 CR6C5D 44441776 IC50 = 9200 nM T70309 CQM3W5 44441785 IC50 = 2900 nM T70309 C0AUC5 44441787 IC50 = 4000 nM T70309 C2LB6P 44441791 IC50 = 4700 nM T70309 C7LR9G 44441793 IC50 = 4700 nM T70309 CBYI82 46905116 Ki = 0.4 nM T70309 CDW32B 71716701 IC50 = 2700 nM T70309 CZ1K2O 127028927 IC50 = 547 nM T70309 CX19MQ 155547708 IC50 = 1300 nM T70309 D00IFJ 10081476 IC50 = 298 nM T70309 D02JEZ 5281426 IC50 > 20 ug.mL-1 T70309 D02ZRX 12012176 IC50 = 2477 nM T70309 D05ZPJ 6917653 IC50 = 1.7 nM T70309 D07KDB 12969973 IC50 = 1400 nM T70309 D08SPJ 10442752 IC50 = 5130 nM T70309 D09KZA 10017278 IC50 = 302 nM T70309 D0H7NB 12012178 IC50 = 3360 nM T70309 D0JH9F 12012177 IC50 = 1690 nM T70309 D0M7OP 10106832 Ki = 9 nM T35842 D0H7AR 70684954 Ki = 8900 nM T35842 D0X9PF 9941379 EC50 = 0.0955 nM T35842 CL04VQ 910537 Ki > 1000000 nM T35842 C0DA9X 2163781 Ki = 32000 nM T35842 CK4YT2 2817655 Ki > 1000000 nM T35842 CB9A2M 2852098 Ki = 16000 nM T35842 C6PQK0 5311058 EC50 = 100 nM T35842 CY60AZ 6918813 EC50 = 350 nM T35842 C2BQE1 6918814 Ki = 4200 nM T35842 CK83QR 6918844 Ki = 1000 nM T35842 CLV3C7 6918849 IC50 = 980 nM T35842 C5U7CS 6918850 Ki = 5700 nM T35842 C0Q5JL 6918851 EC50 = 160000 nM T35842 CRG04O 6918857 Ki = 5800 nM T35842 CM02VS 9808801 EC50 = 420 nM T35842 CKCF18 9867330 EC50 = 2000 nM T35842 CM3Y5H 9893728 IC50 > 10000 nM T35842 CZ5E2C 9915636 Ki = 1300 nM T35842 CCL2T8 9915813 EC50 = 28 nM T35842 CNF37L 9919056 EC50 = 1300 nM T35842 C97MRJ 9960253 Ki = 12000 nM T35842 CLXA58 10025669 Ki = 630.96 nM T35842 C8KI2R 10033237 Ki = 0.17 nM T35842 CZ78WX 10077258 EC50 = 540 nM T35842 C8MCA1 10077773 Ki = 5200 nM T35842 CFX6U7 10123761 EC50 = 50 nM T35842 CFZ5I6 10210964 IC50 = 1400 nM T35842 C8PA3J 10211466 Ki = 20000 nM T35842 C1VCQ8 10213106 IC50 = 4700 nM T35842 CTO7I8 10232787 Ki = 6000 nM T35842 CSNY06 10257242 EC50 = 890 nM T35842 C6Y1ER 10257541 Ki = 2000 nM T35842 CX29KB 10282847 IC50 = 620 nM T35842 C4SCW2 10283036 Ki = 7000 nM T35842 CV3ZJ5 10304463 Ki = 7000 nM T35842 CU13DH 10304547 IC50 = 530 nM T35842 C1E3PC 10304776 IC50 = 220 nM T35842 CT9AR6 10325955 Ki = 4000 nM T35842 C84RZU 10373417 EC50 = 940 nM T35842 C1N3MA 10392968 IC50 = 9100 nM T35842 CPL02I 10463896 EC50 = 2.61 nM T35842 CTEB92 10483153 EC50 = 260 nM T35842 C3NWO8 10484741 EC50 = 13 nM T35842 CBXU29 10510272 EC50 = 0.06 nM T35842 CDC75A 10510273 EC50 = 3 nM T35842 CG3HP6 10534100 EC50 = 6.25 nM T35842 C1IU4G 10534101 EC50 = 2 nM T35842 C8RME3 10606077 EC50 = 0.3 nM T35842 CKNU02 10724780 EC50 = 0.06 nM T35842 CGIC31 10918643 IC50 > 10000 nM T35842 C7IJV5 11038873 EC50 = 1.5 nM T35842 CO2U6S 11156852 Ki = 27 nM T35842 C3V7DK 11180881 Ki = 2300 nM T35842 CHC51K 11181804 Ki = 6000 nM T35842 CUC85X 11215553 EC50 = 228 nM T35842 CF7VQ4 11226756 Ki > 20000 nM T35842 C1T3VM 11249545 Ki = 360 nM T35842 CJ7OT2 11296600 Ki = 1500 nM T35842 C9XBQ7 11308054 Ki > 5000 nM T35842 CS7K4R 11341045 Ki = 400 nM T35842 CU6Y1Z 11341046 Ki = 1900 nM T35842 CY8AJ5 11512024 EC50 = 50.12 nM T35842 CA5GQ7 11592389 EC50 = 22.39 nM T35842 C24UQH 11599302 EC50 = 2951.21 nM T35842 CR0N5C 11613526 EC50 = 29.51 nM T35842 C7F9XQ 11613741 EC50 = 1.585 nM T35842 COLB48 11627577 EC50 = 707.95 nM T35842 CRE2X6 11635051 EC50 = 186.21 nM T35842 C7JU6O 11635265 EC50 = 14.13 nM T35842 CPM61U 11685018 EC50 = 1.585 nM T35842 C3XN4O 11692334 EC50 = 1.585 nM T35842 C6WAM2 11706338 EC50 = 52.48 nM T35842 CH7TQ6 11753695 EC50 = 1020 nM T35842 C7H0ZA 11763303 EC50 = 400 nM T35842 C2SHV7 11786860 Ki = 2100 nM T35842 CS3KM2 11804174 EC50 = 6.25 nM T35842 C0OIV9 11813437 EC50 = 2.5 nM T35842 C7NL4J 11845272 Ki = 42 nM T35842 C4XF1I 11845276 EC50 = 585 nM T35842 CT1F9R 11845438 EC50 = 539 nM T35842 CC42HM 11845440 EC50 = 104 nM T35842 CFKN79 11845444 Ki = 1687 nM T35842 C3JV7M 11845450 EC50 = 0.045 nM T35842 C8WJ6E 11845630 EC50 = 1815 nM T35842 CI1VU0 11845804 Ki = 4.7 nM T35842 C4V9DO 11845813 EC50 = 151 nM T35842 CSZX65 11846669 EC50 = 30 nM T35842 C5HFB2 11846673 EC50 = 232 nM T35842 C25KCW 11846844 EC50 = 71 nM T35842 CO3H9V 11847001 EC50 = 1220 nM T35842 CECQ63 11847312 EC50 = 390 nM T35842 CT4EC3 11966875 EC50 = 1428 nM T35842 CI9W3G 15953833 IC50 = 230 nM T35842 C2BLT4 16007263 EC50 = 526 nM T35842 CK3T2B 16038121 EC50 = 135 nM T35842 C4N0VF 16046215 Ki = 3100 nM T35842 CX68DN 16049796 EC50 > 10000 nM T35842 C8UXP9 16126683 EC50 = 31.8 nM T35842 CPTO16 16132144 EC50 = 0.091 nM T35842 C25XZF 17880880 Ki > 1000000 nM T35842 CU19BT 24740419 Ki = 6400 nM T35842 CD90WZ 24740655 Ki = 8400 nM T35842 C5TA3W 24774358 IC50 > 10000 nM T35842 CO4JK2 24774437 EC50 > 1000 nM T35842 CMB27G 24774521 IC50 > 10000 nM T35842 C2TAK6 24774601 IC50 > 10000 nM T35842 C2A1SX 24848995 EC50 > 3000 nM T35842 CZT4J0 24858627 IC50 > 1500 nM T35842 CB9M3F 24873537 Ki = 3350 nM T35842 CS0L2N 24882666 Ki > 25000 nM T35842 CJ5HN6 25128748 EC50 = 2300 nM T35842 C3WE0T 25128749 EC50 = 1076 nM T35842 CP5TN2 25128751 EC50 = 878 nM T35842 CUTA14 25129105 EC50 = 193 nM T35842 CPL49Z 25129107 EC50 = 145 nM T35842 C4N5DH 25129108 EC50 = 44 nM T35842 CDC2Q6 25129109 EC50 = 50 nM T35842 CVSO97 25129453 EC50 = 80 nM T35842 CE79VX 25131477 Ki = 16832 nM T35842 C1B7KF 25131478 Ki = 63 nM T35842 CIJ6P4 25132524 EC50 = 1697 nM T35842 CY42MT 25132525 EC50 = 1523 nM T35842 C9QG3J 25132526 EC50 = 796 nM T35842 CL3JV6 25132864 EC50 = 308 nM T35842 C57QZT 25132866 EC50 = 432 nM T35842 CR6YZ2 25132867 EC50 = 392 nM T35842 C8AO5Y 25133207 EC50 = 734 nM T35842 C3VGX6 25133208 EC50 = 48 nM T35842 C3KRA8 25133209 EC50 = 98 nM T35842 C9U6CQ 25133210 EC50 = 170 nM T35842 C74ACT 25133556 EC50 = 10 nM T35842 CW7O1N 25133903 Ki = 4469 nM T35842 CG3R0Y 25133907 EC50 = 1505 nM T35842 C4HK6C 42630327 EC50 = 0.263 nM T35842 CU4S6X 44157099 IC50 = 1.2 nM T35842 CIOF26 44158168 EC50 = 820 nM T35842 C53LJK 44158169 EC50 = 2700 nM T35842 CF7X1N 44158255 EC50 = 19000 nM T35842 CF6PT4 44158337 EC50 = 620 nM T35842 CHKI60 44265225 Ki > 1000000 nM T35842 CXN2R4 44265309 Ki > 1000000 nM T35842 C3EJ1R 44265312 Ki = 26000 nM T35842 CWPT03 44265315 Ki = 9800 nM T35842 CJ1M6N 44265347 Ki = 27000 nM T35842 CEQ6K7 44265351 Ki = 46000 nM T35842 CSL48C 44265374 Ki = 1500 nM T35842 C97AIK 44265472 Ki = 12000 nM T35842 CLE96R 44265479 Ki > 1000000 nM T35842 CV8GX6 44265487 Ki = 19000 nM T35842 C2CPG9 44265489 Ki = 28000 nM T35842 CLP5G3 44265496 Ki = 630.96 nM T35842 C51TPY 44265586 Ki > 1000 nM T35842 CH5WM7 44265588 Ki > 1000 nM T35842 CT89LY 44265589 Ki = 29000 nM T35842 CZS3C7 44265590 Ki > 1000000 nM T35842 C3YKG9 44265591 Ki = 32000 nM T35842 C74SBD 44265625 Ki > 1000 nM T35842 CRQ92O 44265626 Ki > 1000 nM T35842 CT2S8I 44265639 Ki = 1300 nM T35842 C18JZD 44265656 Ki > 1000000 nM T35842 CZWE24 44265658 Ki = 4500 nM T35842 CD8UC0 44265662 Ki > 1000 nM T35842 C6OU7D 44265665 Ki > 1000 nM T35842 CC28FH 44265672 Ki = 2200 nM T35842 CSK9V6 44265674 Ki > 1000 nM T35842 CS46LN 44265675 Ki > 1000000 nM T35842 C9E0TB 44265681 Ki = 2900 nM T35842 CCGI15 44265707 Ki = 5900 nM T35842 CION54 44265708 Ki = 26000 nM T35842 C9CM8W 44265711 Ki = 15000 nM T35842 CP1E6X 44265715 Ki = 2900 nM T35842 CRFQ64 44265719 Ki = 74000 nM T35842 CXUI50 44265722 Ki = 22000 nM T35842 CVEG42 44265727 Ki > 1000 nM T35842 CC4S8V 44265739 Ki > 1000 nM T35842 CG1CH0 44265748 Ki > 1000 nM T35842 C82FPN 44265749 Ki = 8700 nM T35842 C05MIH 44265751 Ki = 3981.07 nM T35842 CP82FI 44265757 Ki > 1000 nM T35842 CE6A0Z 44265759 Ki > 1000 nM T35842 CPE83Q 44269189 EC50 = 0.35 nM T35842 CCP5L2 44269214 EC50 = 3.8 nM T35842 CN5TI2 44269217 EC50 = 0.19 nM T35842 C4M2LJ 44269245 EC50 = 220 nM T35842 C29BRD 44269246 EC50 = 510 nM T35842 C6LD9E 44275119 EC50 = 1275 nM T35842 CFIT54 44275175 EC50 = 1330 nM T35842 CA7DX2 44275263 IC50 = 5815 nM T35842 CB4WG5 44275265 EC50 = 140 nM T35842 C3SH7Q 44275312 IC50 = 14790 nM T35842 CIA54K 44275371 EC50 = 480 nM T35842 CBS9X6 44275372 EC50 = 480 nM T35842 CBW0I1 44275650 EC50 = 0.4 nM T35842 CO9BJ6 44275654 EC50 = 370 nM T35842 COUM34 44275656 EC50 = 12 nM T35842 CSI8T3 44277299 EC50 = 990 nM T35842 CCGT80 44277300 EC50 = 1480 nM T35842 CLG8Y1 44277301 EC50 = 890 nM T35842 C3PQM1 44277422 EC50 = 3380 nM T35842 CD54ZT 44277558 EC50 = 1710 nM T35842 C5OHC4 44277696 EC50 = 10 nM T35842 CMU9P1 44278071 EC50 = 230 nM T35842 C9Y7KM 44278193 EC50 = 295 nM T35842 CBWJ71 44278194 EC50 = 195 nM T35842 COS0B2 44278195 EC50 = 1220 nM T35842 C8A1GE 44278223 EC50 = 680 nM T35842 C9BR8N 44285017 IC50 = 500 nM T35842 C6RDN1 44285101 EC50 = 1 nM T35842 C1B3JD 44285102 EC50 = 10000 nM T35842 C86RFZ 44285133 EC50 = 0.1 nM T35842 COS13M 44285136 EC50 = 1000 nM T35842 C0JO7K 44285147 IC50 = 500 nM T35842 CCG7U0 44285223 IC50 = 1000 nM T35842 C76VJU 44285234 EC50 = 30 nM T35842 C51VFH 44285236 EC50 = 3000 nM T35842 C0XN3K 44285237 EC50 = 0.1 nM T35842 C2Y9AV 44285238 EC50 = 100 nM T35842 CIA4M6 44285239 EC50 = 5000 nM T35842 C5L3QZ 44285261 EC50 = 10 nM T35842 C6FZQ3 44285262 IC50 = 500 nM T35842 C4IK2Q 44285313 IC50 = 100 nM T35842 C7BM6H 44285368 IC50 = 1000 nM T35842 CZ3D0Y 44285388 EC50 = 100 nM T35842 CTQ9E3 44285416 EC50 = 10000 nM T35842 CEA3Q9 44285417 EC50 = 0.3 nM T35842 CED1W0 44285432 EC50 = 1000 nM T35842 CU8PH5 44293516 IC50 = 1.94 nM T35842 C7DZ1Q 44293599 EC50 = 34.2 nM T35842 C57HNX 44307979 IC50 > 10000 nM T35842 C8LZV7 44308004 IC50 > 10000 nM T35842 CFP7W8 44308044 IC50 > 10000 nM T35842 C79WRA 44308214 IC50 > 10000 nM T35842 CT76SR 44308215 IC50 > 10000 nM T35842 C3U0CW 44317053 EC50 = 1700 nM T35842 CKH3J2 44317070 EC50 = 350 nM T35842 CU0FY3 44317071 EC50 = 255 nM T35842 CAW8L7 44317241 EC50 = 10 nM T35842 CK7LG6 44317242 EC50 = 950 nM T35842 CZTI78 44317254 EC50 = 1 nM T35842 CVW5B7 44317276 EC50 = 15 nM T35842 C4ZST8 44317277 EC50 = 85 nM T35842 C90PCI 44317278 EC50 = 60 nM T35842 CLO83G 44317279 EC50 = 900 nM T35842 CQ59BO 44320339 Ki = 1584.89 nM T35842 C6UML0 44322786 EC50 = 88 nM T35842 C3CL8S 44322787 EC50 = 8 nM T35842 C5SZ6K 44322788 EC50 = 7.5 nM T35842 C9HQ8Z 44322812 EC50 = 3.5 nM T35842 CJD5K7 44322895 EC50 = 2 nM T35842 CSH73B 44322896 Ki = 0.006 nM T35842 C3V7PO 44322923 EC50 = 8 nM T35842 CA9F8I 44322924 EC50 = 7 nM T35842 C32ADM 44322957 EC50 = 6.5 nM T35842 CU1R6F 44322958 EC50 = 5 nM T35842 CPG80V 44322959 EC50 = 2 nM T35842 CJ73UR 44322977 EC50 = 7 nM T35842 CW5T8L 44322986 EC50 = 7 nM T35842 CN12SY 44322987 EC50 = 4.5 nM T35842 C8W2GN 44322994 EC50 = 9.5 nM T35842 CEV0F8 44323015 EC50 = 9 nM T35842 CSL38N 44323016 EC50 = 33.3 nM T35842 CI70FV 44323029 Ki = 3.5 nM T35842 CNB32J 44323031 EC50 = 0.5 nM T35842 CP9FE1 44323032 EC50 = 2 nM T35842 CCX5N0 44323033 EC50 = 6.8 nM T35842 C7RT2W 44323034 EC50 = 13.7 nM T35842 CTUP81 44325899 EC50 = 3.33 nM T35842 C8BID0 44325926 EC50 = 0.19 nM T35842 C5NY9A 44325927 EC50 = 1 nM T35842 C9MA4R 44343337 EC50 = 0.016 nM T35842 CD9ER8 44343341 EC50 = 0.036 nM T35842 C46OFK 44343362 EC50 = 0.055 nM T35842 CL8Y3V 44343363 EC50 = 0.005 nM T35842 C6E7SA 44349019 EC50 > 3000 nM T35842 C8EA5J 44355350 EC50 = 0.055 nM T35842 C2QW1I 44364160 EC50 = 70 nM T35842 C61CYL 44372908 EC50 = 55 nM T35842 CWT5B7 44372933 EC50 = 10 nM T35842 C8D1MC 44372942 EC50 = 180 nM T35842 CEW35X 44372964 EC50 = 611 nM T35842 C2UCY5 44373177 EC50 = 20 nM T35842 CZ42QB 44373197 EC50 = 0.4 nM T35842 CCB05K 44373198 EC50 = 54 nM T35842 CX92FV 44373317 EC50 = 274 nM T35842 CNDX59 44379584 IC50 = 637 nM T35842 CUEW16 44379585 IC50 = 10000 nM T35842 C8V4YU 44379727 EC50 = 313 nM T35842 C8MY6B 44379728 EC50 = 31 nM T35842 CKN48P 44379730 EC50 = 2700 nM T35842 C1LP6F 44379745 EC50 = 825 nM T35842 CZDA19 44379746 IC50 = 1500 nM T35842 CRK73M 44379968 EC50 = 5200 nM T35842 C0F8NW 44379982 IC50 = 440 nM T35842 CBNO94 44379988 EC50 = 510 nM T35842 C8L7SA 44379989 EC50 = 60 nM T35842 CI91UV 44380006 EC50 = 23 nM T35842 C8BX4R 44380007 EC50 = 2 nM T35842 C80ZVG 44380208 IC50 = 8200 nM T35842 C7Y3DT 44380209 EC50 = 60 nM T35842 CD8HL0 44392514 Ki = 2200 nM T35842 CE21OM 44392535 Ki = 530 nM T35842 C3IHV4 44393417 Ki = 2000 nM T35842 C2J1ML 44393418 Ki = 3200 nM T35842 CQ3L0D 44393421 Ki = 11000 nM T35842 C9C7SD 44393430 Ki = 152000 nM T35842 C47HVD 44393441 Ki = 13000 nM T35842 C1OG5U 44393450 Ki = 36000 nM T35842 CK5D8I 44394079 Ki = 42 nM T35842 C25TVF 44394093 EC50 = 555 nM T35842 C5K7CG 44394580 EC50 = 565 nM T35842 C08QML 44394581 EC50 = 536 nM T35842 C0OMU3 44394582 EC50 = 441 nM T35842 CL3P2Q 44394583 EC50 = 381 nM T35842 C5SGR6 44394584 EC50 = 1214 nM T35842 CLXA10 44394585 EC50 = 856 nM T35842 C48NFW 44394586 EC50 = 502 nM T35842 C8GUD1 44394622 EC50 = 13 nM T35842 C9O4GM 44394623 EC50 = 0.009 nM T35842 C29ELZ 44394624 EC50 = 0.05 nM T35842 CP4A0B 44394625 EC50 = 867 nM T35842 C94PGA 44394626 EC50 = 1982 nM T35842 CF4O9U 44394627 EC50 = 803 nM T35842 CZ37TO 44394654 EC50 = 378 nM T35842 CPE65R 44394655 EC50 = 211 nM T35842 C9LKB5 44394656 EC50 = 1028 nM T35842 CG1Q8L 44394657 EC50 = 499 nM T35842 CHG12Y 44394658 EC50 = 349 nM T35842 C9OTX4 44394659 EC50 = 567 nM T35842 CNHD57 44394660 EC50 = 597 nM T35842 CHTM92 44394689 EC50 = 1430 nM T35842 C04RCL 44394690 EC50 = 947 nM T35842 CT9D5Y 44394691 EC50 = 577 nM T35842 CHDB95 44394692 EC50 = 541 nM T35842 CHZF38 44394693 EC50 = 699 nM T35842 C9Y6ZI 44394694 EC50 = 442 nM T35842 C06PXF 44394695 EC50 = 113 nM T35842 CJ97VD 44394730 EC50 = 600 nM T35842 C1IE7P 44394731 EC50 = 848 nM T35842 CLF0X5 44394732 EC50 = 2162 nM T35842 C9QR1L 44394733 EC50 = 505 nM T35842 CP1IR5 44394734 EC50 = 700 nM T35842 C2UY8G 44394735 EC50 = 892 nM T35842 CTY36S 44394736 EC50 = 671 nM T35842 CR5B6L 44394748 EC50 = 2157 nM T35842 CW13LR 44394749 EC50 = 785 nM T35842 CL3A0O 44394750 EC50 = 1894 nM T35842 CIGZ40 44394783 EC50 = 144 nM T35842 C62FUR 44394784 EC50 = 23 nM T35842 CCZ37I 44394785 EC50 = 114 nM T35842 C8RHG3 44394786 EC50 = 41 nM T35842 CQD01R 44394787 EC50 = 841 nM T35842 CO43JY 44394788 EC50 = 985 nM T35842 CCE30Z 44394789 EC50 = 534 nM T35842 CVUQ61 44395681 Ki = 1200 nM T35842 CZ2C9L 44397028 Ki = 2800 nM T35842 CDZ3O4 44397030 Ki = 4600 nM T35842 CX07ID 44397304 Ki = 4500 nM T35842 C6F0QR 44397455 IC50 = 940 nM T35842 C61RQJ 44400934 Ki = 6800 nM T35842 C2IJZ5 44400935 Ki = 6900 nM T35842 CYF7N9 44401275 Ki > 5000 nM T35842 CKH54Y 44401285 Ki > 5000 nM T35842 C1JK9O 44401341 Ki > 5000 nM T35842 CTOS16 44401367 Ki > 5000 nM T35842 C3S2XK 44401371 Ki > 5000 nM T35842 CH1OX7 44401386 Ki > 5000 nM T35842 CR8GT9 44401392 Ki > 5000 nM T35842 CBQ7N3 44401418 Ki > 5000 nM T35842 C1O0YW 44401421 Ki > 5000 nM T35842 CJNH94 44401440 Ki > 5000 nM T35842 CGA3W5 44401462 Ki > 5000 nM T35842 CUZJ52 44401513 Ki > 5000 nM T35842 C9Y0LO 44401553 Ki > 5000 nM T35842 C7E3YU 44401573 Ki > 5000 nM T35842 C5LID4 44401581 Ki > 5000 nM T35842 CGNC86 44401587 Ki > 5000 nM T35842 C74QHS 44401592 Ki > 5000 nM T35842 CX30HI 44401607 Ki > 5000 nM T35842 C1CY7E 44404525 EC50 = 1300 nM T35842 CUZ2B7 44404526 EC50 = 690 nM T35842 C3I9PN 44404527 EC50 = 210 nM T35842 CNH3C0 44404528 EC50 = 1300 nM T35842 CH5E4L 44405832 EC50 = 2900 nM T35842 CRMV98 44408154 EC50 = 460 nM T35842 CIWX60 44408155 EC50 = 1500 nM T35842 COG72Y 44408173 EC50 = 680 nM T35842 C3CQ4J 44408189 EC50 = 950 nM T35842 CW08ZJ 44408190 EC50 = 1300 nM T35842 CNWJ27 44408252 EC50 = 980 nM T35842 CH68SP 44408253 EC50 = 970 nM T35842 CCFV91 44408275 EC50 = 2100 nM T35842 CZ3YG9 44408276 EC50 = 2600 nM T35842 CAFP51 44408286 EC50 = 550 nM T35842 CR8HZ7 44408287 EC50 = 1300 nM T35842 COC7D2 44408388 EC50 = 1700 nM T35842 CJ4N3I 44409103 Ki = 9 nM T35842 C2NJ0V 44409104 Ki = 30 nM T35842 CKF52N 44409140 Ki = 3992 nM T35842 C5XEI8 44409206 Ki = 71 nM T35842 C9EXZ2 44409337 Ki = 8562 nM T35842 CFT41O 44409338 Ki = 22267 nM T35842 CUB1Q2 44409339 Ki = 23400 nM T35842 CK5GO1 44409379 Ki = 12288 nM T35842 C48WZD 44410802 Ki = 8600 nM T35842 C43IKV 44410803 Ki = 3000 nM T35842 CW6ZC0 44413576 EC50 = 3301.8 nM T35842 C24AUD 44413828 EC50 = 72 nM T35842 C08PBM 44413829 EC50 = 28 nM T35842 CT4FW5 44413830 EC50 = 4.3 nM T35842 C8IDV1 44413831 EC50 = 1362 nM T35842 CZ3Q4T 44413832 EC50 = 1070 nM T35842 CV6Z8C 44413842 EC50 = 521 nM T35842 C4P0LS 44413879 EC50 = 3 nM T35842 C84OJQ 44413880 Ki = 15 nM T35842 CN7I2S 44413881 EC50 = 1337 nM T35842 CF6O4K 44413913 EC50 = 328 nM T35842 CS42BM 44413914 EC50 = 0.3 nM T35842 CN18BL 44413930 Ki = 85 nM T35842 C4BMF6 44413931 Ki = 35 nM T35842 C9WNH8 44413932 EC50 = 52 nM T35842 CKZ86P 44413938 Ki = 182 nM T35842 CL2RK9 44413968 Ki = 19 nM T35842 CM2J9Z 44413969 Ki = 340 nM T35842 C34XGB 44413970 EC50 = 402 nM T35842 C3KQ8H 44415912 EC50 = 317 nM T35842 CDN97X 44415913 EC50 = 0.07 nM T35842 CAL83K 44415914 Ki = 1 nM T35842 C5CF0M 44415918 EC50 = 1.7 nM T35842 CXI18W 44415919 Ki = 14 nM T35842 C6DH7I 44415920 EC50 = 3.7 nM T35842 C06CYU 44415956 Ki = 4384 nM T35842 CD2A9T 44415972 Ki = 4058 nM T35842 CHT4E8 44415991 Ki = 5820 nM T35842 CPX62S 44416014 Ki = 21703 nM T35842 C69CUX 44416057 EC50 = 0.37 nM T35842 C56DHI 44416060 EC50 = 104 nM T35842 CB2TU4 44416106 EC50 = 2.3 nM T35842 CP9T4B 44416122 Ki = 2132 nM T35842 C9KLB0 44416135 EC50 = 353 nM T35842 C37XPA 44416152 Ki = 958 nM T35842 C1F7CU 44417402 IC50 > 10000 nM T35842 CD7ZM1 44417550 IC50 = 1000 nM T35842 CBCR82 44417551 IC50 > 1000 nM T35842 CD72MS 44417553 IC50 > 1000 nM T35842 CT58RV 44417554 IC50 = 750 nM T35842 C4G2BZ 44417555 IC50 > 1000 nM T35842 C32QEO 44418413 EC50 > 10000 nM T35842 C7FEU6 44418420 EC50 > 10000 nM T35842 CZW07E 44418421 IC50 = 4 nM T35842 CLQG83 44418430 IC50 = 2.2 nM T35842 C8VG1S 44418431 IC50 = 1.3 nM T35842 C3HPI5 44418437 EC50 > 10000 nM T35842 CMD5N2 44418438 EC50 > 10000 nM T35842 CQE30X 44422937 IC50 = 980 nM T35842 C14FZP 44422938 IC50 > 2000 nM T35842 CE0H3Y 44422957 IC50 > 10000 nM T35842 C6H0NU 44422958 EC50 > 2500 nM T35842 C7I0KW 44422959 IC50 > 10000 nM T35842 C46XOB 44422960 IC50 > 10000 nM T35842 CNM90E 44422961 IC50 > 10000 nM T35842 C2K3BL 44422962 IC50 > 10000 nM T35842 C3E6VO 44422994 EC50 > 500 nM T35842 CHU7G0 44422996 EC50 = 540 nM T35842 C2LQW9 44422997 EC50 = 63 nM T35842 CJM09S 44422998 EC50 = 300 nM T35842 CI9HF1 44422999 EC50 = 5.3 nM T35842 CXH5F8 44423009 EC50 = 1300 nM T35842 C3VOD0 44423010 EC50 = 89 nM T35842 C7UI3W 44423011 EC50 = 880 nM T35842 CI05BD 44423012 EC50 > 2500 nM T35842 C5EJ3P 44423013 IC50 > 10000 nM T35842 C2NR7G 44423014 EC50 = 50 nM T35842 CV3TL5 44423015 EC50 = 60 nM T35842 CN5RD6 44431510 EC50 > 10000 nM T35842 CF3H8A 44431511 EC50 > 10000 nM T35842 CVB07O 44431512 EC50 = 900 nM T35842 CY80GN 44431513 IC50 = 580 nM T35842 COCE51 44431515 EC50 = 0.3 nM T35842 CV62SP 44432932 Ki = 9300 nM T35842 CL3ZR1 44432964 Ki > 10000 nM T35842 C0L4NV 44432966 Ki = 7500 nM T35842 CO93SX 44443035 Ki = 3900 nM T35842 CTP3D6 44453826 EC50 > 50000 nM T35842 C4FV3C 44453850 EC50 > 50000 nM T35842 CEI35V 44453902 EC50 > 25000 nM T35842 CUPG04 44453903 Ki > 10000 nM T35842 C63APB 44456219 Ki = 120 nM T35842 CQ8J9K 44569175 EC50 = 104 nM T35842 CL8GU3 44569176 EC50 = 69 nM T35842 CJ6GZ3 44577063 Ki = 8200 nM T35842 CGTV08 44577094 Ki = 6200 nM T35842 CEJ96P 44577510 EC50 = 2 nM T35842 CRSQ61 44577514 IC50 = 760 nM T35842 C6Y1BS 44577515 IC50 > 2000 nM T35842 CM47HW 44577516 EC50 > 1000 nM T35842 C8B1WR 44577520 EC50 = 71 nM T35842 C9ZD5W 44577522 IC50 > 1000 nM T35842 C3NSW7 44577523 EC50 = 100 nM T35842 CR5ZS2 44583562 EC50 = 760 nM T35842 CWFB17 44583567 EC50 = 1.5 nM T35842 CN7AM1 45487404 EC50 = 5 nM T35842 CJB6H0 46203215 EC50 > 7810 nM T35842 CY12SB 46228659 EC50 = 1548.82 nM T35842 C10VXP 46228660 EC50 = 15.85 nM T35842 C8XUS4 46228689 EC50 = 61.66 nM T35842 C5FVJ9 46228690 EC50 = 1.585 nM T35842 CCK7I1 46228725 EC50 > 30000 nM T35842 CD5Q8V 46228726 EC50 = 295.12 nM T35842 CJ7R0X 46228763 EC50 > 30000 nM T35842 CYD2R3 46228764 EC50 = 35.48 nM T35842 CQ53EA 46228813 EC50 = 177.83 nM T35842 CMX28H 46228814 EC50 = 398.11 nM T35842 C7FAY5 46228815 EC50 = 12.59 nM T35842 C82NVP 46228841 EC50 > 30000 nM T35842 CEDL84 46228842 EC50 = 831.76 nM T35842 CP86QH 46228843 EC50 > 30000 nM T35842 C4BD8Z 46228844 EC50 = 1174.9 nM T35842 CR6PF0 46228845 EC50 = 794.33 nM T35842 CCN14H 46228846 EC50 = 1380.38 nM T35842 C3T1NY 46228847 EC50 > 30000 nM T35842 COW85F 46228848 EC50 > 30000 nM T35842 CZLY24 46228849 EC50 > 30000 nM T35842 C5VAN7 46228850 EC50 > 30000 nM T35842 C0X9KS 46228888 EC50 = 3715.35 nM T35842 CQ28TZ 46884748 EC50 = 620 nM T35842 CD3E4C 46885323 EC50 > 8740 nM T35842 CNW43Y 46885367 EC50 > 4910 nM T35842 CE4SF8 46885368 EC50 = 1100 nM T35842 CV23JL 46885415 EC50 = 350 nM T35842 CHPS01 46885417 EC50 > 11900 nM T35842 C4SVE1 46885480 EC50 > 16700 nM T35842 C5QI7J 46885481 EC50 > 8220 nM T35842 COU5X2 46885482 EC50 > 3070 nM T35842 CG9NJ1 46885523 EC50 = 1850 nM T35842 CS90MN 46885524 EC50 = 3900 nM T35842 CQ94VM 46885526 EC50 > 16700 nM T35842 C90ABZ 46885558 EC50 > 9000 nM T35842 C0MI3C 46885560 EC50 > 10000 nM T35842 C0Y9NF 46885711 EC50 > 5880 nM T35842 C3O5BR 46885712 EC50 = 1120 nM T35842 CG6XN0 46885759 EC50 > 6470 nM T35842 CK8D6G 46885760 EC50 > 5010 nM T35842 C0C8GN 46885761 EC50 = 6570 nM T35842 CY30PG 46885815 EC50 = 1170 nM T35842 CEA70O 46885816 EC50 = 3610 nM T35842 CWN89S 46885863 EC50 > 6150 nM T35842 C8UTI7 46885907 EC50 > 8250 nM T35842 CFC5L1 46885972 EC50 = 750 nM T35842 CO3S1Q 46905544 Ki > 5000 nM T35842 C96XEU 46905545 Ki > 5000 nM T35842 C1EMQ2 49861348 EC50 = 1020 nM T35842 C9QU3G 49862375 EC50 = 1200 nM T35842 CPZI97 49862377 EC50 = 520 nM T35842 CY7R2T 49862378 EC50 = 560 nM T35842 C7GA4I 49862425 IC50 = 5000 nM T35842 C0QD9I 51346770 EC50 = 16 nM T35842 C30PGL 51346771 EC50 = 12 nM T35842 CBQN64 52918026 IC50 = 5100 nM T35842 C5RGD8 52943036 EC50 = 158.49 nM T35842 CG5TJ0 53240339 EC50 = 26 nM T35842 CDKP06 54580990 IC50 > 4000 nM T35842 C6GET3 54582029 IC50 > 4000 nM T35842 CQ7O3U 54584301 EC50 = 910 nM T35842 C8PIL3 54584302 EC50 = 250 nM T35842 CN6F2C 54586246 EC50 = 400 nM T35842 CEU0M6 54587278 EC50 = 280 nM T35842 CTSB57 56850936 Ki = 1.8 nM T35842 C1U2DB 56851057 Ki = 0.24 nM T35842 C2WAO4 57634921 Ki = 200 nM T35842 C4VT5C 57634925 Ki = 73 nM T35842 CKW2T0 57646411 Ki = 3.2 nM T35842 C8F5XG 57646441 Ki = 8 nM T35842 CH1LU3 58777892 Ki = 4000 nM T35842 CS27GN 70682904 Ki = 45000 nM T35842 C73SKU 70682946 IC50 = 1 nM T35842 CPJ08L 70688853 Ki = 130 nM T35842 CE28CX 70691332 EC50 = 0.036 nM T35842 C3G7MZ 70695694 EC50 = 110 nM T35842 CF4LE6 71449181 EC50 = 0.2 nM T35842 CBP20G 71452716 EC50 = 14 nM T35842 CEB0P9 71452732 Ki = 7000 nM T35842 CY16AM 71454518 Ki = 1500 nM T35842 CE83FK 71454570 EC50 = 0.44 nM T35842 CQPB08 71456236 EC50 = 0.1 nM T35842 CNRV69 71456245 EC50 = 240 nM T35842 C09YUJ 71456276 EC50 = 0.02 nM T35842 CA5GY9 71458041 EC50 = 4 nM T35842 CU17GR 71458055 Ki = 20000 nM T35842 C6YR0U 71458117 IC50 > 10000 nM T35842 C3V0DA 71459896 EC50 = 830 nM T35842 CJ52CU 71459938 EC50 = 220 nM T35842 C12JDC 71461643 EC50 = 1 nM T35842 CECQ16 71461657 Ki = 3000 nM T35842 C24GWM 71461662 Ki = 11000 nM T35842 CZ94CM 71461730 EC50 = 0.098 nM T35842 CYA8G1 71717886 EC50 = 55 nM T35842 CG3H2F 73345549 EC50 = 48 nM T35842 C1A5SK 73345616 IC50 = 2900 nM T35842 CI0DV9 73345617 IC50 > 5000 nM T35842 CD1NE3 73345618 IC50 = 1300 nM T35842 C38VZT 73347097 EC50 = 23 nM T35842 C31UAJ 73347130 EC50 = 420 nM T35842 C7DYR4 73347133 EC50 = 3 nM T35842 CZ91TE 73347138 EC50 = 3.3 nM T35842 CK46SP 73347139 EC50 > 2500 nM T35842 CX9LF8 73347140 IC50 > 1000 nM T35842 CW8F4U 73348170 EC50 = 0.3 nM T35842 C4SR8Z 73348617 EC50 = 2 nM T35842 CK69FV 73348634 EC50 = 5 nM T35842 C82VMG 73350129 EC50 = 0.3 nM T35842 CI9FS8 73350149 EC50 = 30 nM T35842 CI07CR 73350214 EC50 = 735 nM T35842 CMLR03 73350220 EC50 = 28 nM T35842 CKWH98 73351727 EC50 = 130 nM T35842 CWHE24 73351850 EC50 = 150 nM T35842 C1L7HK 73353100 IC50 = 0.3 nM T35842 C8C0LW 73353205 EC50 = 330 nM T35842 CGVC68 73353206 IC50 > 1000 nM T35842 CV27XE 73353216 EC50 = 4380 nM T35842 CA4MR1 73354641 EC50 = 10 nM T35842 CT71MQ 73354672 EC50 > 10000 nM T35842 C15BNT 73354704 EC50 = 900 nM T35842 C0ISQ4 73354708 EC50 = 350 nM T35842 CJS25D 73354709 EC50 > 500 nM T35842 C7OL2D 73354716 EC50 = 830 nM T35842 C5XHR6 73354758 IC50 = 1000 nM T35842 CCS79L 73354761 IC50 = 1000 nM T35842 C7OT4D 73354780 EC50 = 0.1 nM T35842 C6L8AD 101043841 EC50 = 860 nM T35842 C1KS2F 101043843 EC50 = 940 nM T35842 CDBN30 118718826 EC50 = 0.005 nM T35842 CCL46X 118718855 IC50 > 10000 nM T35842 CK6FL5 118718881 EC50 = 0.3 nM T35842 C8ME0B 118735099 IC50 = 1352 nM T35842 CK17XF 118735100 EC50 = 226 nM T35842 C1O7GU 118735101 EC50 = 700 nM T35842 CBTC79 118735102 EC50 = 1000 nM T35842 C1O3GL 118735103 EC50 = 750 nM T35842 C65WMB 122184498 EC50 = 3.3 nM T35842 CH9L8O 122184499 EC50 = 5 nM T35842 CAQ17N 122184571 IC50 = 192 nM T35842 CK48WX 122184572 EC50 = 50.8 nM T35842 CF9PO7 122184573 EC50 = 2210 nM T35842 C3FBZ9 122184574 IC50 = 106 nM T35842 CCP0X7 122184575 EC50 = 36 nM T35842 C7OBX1 122184576 EC50 = 2.1 nM T35842 CU73AF 122184577 EC50 = 563 nM T35842 CGB7F4 122184578 IC50 = 196 nM T35842 CB7HZ8 122184579 IC50 = 111 nM T35842 C9HE4L 122184580 IC50 = 916 nM T35842 C9MJT7 122184581 IC50 = 1050 nM T35842 C20NAY 122184582 EC50 = 759 nM T35842 CH1B8W 122184631 EC50 = 3.7 nM T35842 CLXB63 122184632 IC50 = 2520 nM T35842 CIJ14O 122184633 IC50 = 246 nM T35842 CDSR31 122184634 EC50 = 214 nM T35842 CL28BX 122184635 IC50 = 242 nM T35842 CYOR02 122184636 IC50 = 256 nM T35842 C09LFS 122184637 EC50 = 23 nM T35842 C5CDX9 122184638 IC50 = 824 nM T35842 C64BPZ 122184639 EC50 = 276 nM T35842 CEDT39 122184640 EC50 = 1970 nM T35842 CLB43S 122184641 EC50 = 117 nM T35842 CN4L5U 122184908 EC50 = 366 nM T35842 CG0U7B 122184909 EC50 = 841 nM T35842 CZ4HW7 122184910 EC50 = 20 nM T35842 C6KW7J 122184911 EC50 = 58 nM T35842 CK3VM5 122184912 EC50 = 273 nM T35842 C0AFH9 122184913 EC50 = 679 nM T35842 CNBA05 122184914 EC50 = 25.7 nM T35842 C7CLU6 133053557 EC50 = 28 nM T35842 CJNF06 137631599 EC50 = 4.074 nM T35842 COM8N7 137631628 IC50 = 137 nM T35842 CW9P1D 137633115 EC50 = 40 nM T35842 CTD90C 137634090 EC50 = 1400 nM T35842 CU4KL7 137636677 EC50 = 29.51 nM T35842 CVC3Q2 137636965 EC50 = 389.05 nM T35842 CMJ4I7 137637705 IC50 = 16 nM T35842 C2FEA6 137638725 EC50 = 97.72 nM T35842 CZ74WU 137639140 EC50 = 4500 nM T35842 CKR14I 137639770 EC50 = 0.7 nM T35842 CHB9X0 137640703 EC50 = 5.754 nM T35842 CBL5Z9 137641157 EC50 = 3.548 nM T35842 CCPD94 137641398 EC50 = 0.7413 nM T35842 CTN96O 137642298 EC50 = 4.5 nM T35842 CAT50J 137643076 EC50 = 8 nM T35842 C5R2TI 137643266 EC50 = 31 nM T35842 CJ1I7B 137645567 EC50 > 1000 nM T35842 CKES17 137646333 EC50 = 3467.37 nM T35842 CT18GM 137646617 EC50 = 1318.26 nM T35842 CY7K4J 137647538 EC50 = 0.5248 nM T35842 C5X7AK 137648344 IC50 = 1.1 nM T35842 CF3VP0 137651074 EC50 = 4.6 nM T35842 CF5Z2W 137653739 EC50 = 0.01 nM T35842 CKX3Q9 137653925 EC50 = 416.87 nM T35842 CMO01K 137655905 EC50 = 41.69 nM T35842 CJ9RO7 137657609 EC50 > 1000 nM T35842 C5FI6X 137657633 EC50 = 70 nM T35842 COS0A1 137658158 EC50 = 54.95 nM T35842 CS1PR7 137659394 EC50 = 38.02 nM T35842 CHB32J 137659790 EC50 = 85.11 nM T35842 CQ7S0L 137659949 Ki = 30 nM T35842 C2XLI7 137660671 EC50 = 0.9333 nM T35842 C98FVD 137660993 EC50 = 1.514 nM T35842 C2WC5J 145948876 EC50 > 1000 nM T35842 CUC3S2 145948912 EC50 = 26 nM T35842 C8D7OM 145964017 EC50 = 16 nM T35842 CCK75J 145964837 EC50 = 67 nM T35842 CS73TM 145966364 EC50 = 8.6 nM T35842 CHU51B 145966490 EC50 = 15 nM T35842 CJO1Y6 145966716 EC50 = 48 nM T35842 C9RA7Q 145967155 EC50 = 41 nM T35842 CICD84 145971389 EC50 = 25 nM T35842 C97DEG 145971673 EC50 = 60 nM T35842 CEV4F6 145972289 EC50 = 108 nM T35842 C9NRU8 145973779 EC50 = 631 nM T35842 CYD0J5 145973975 EC50 = 14 nM T35842 CR2NQ5 145975465 EC50 = 87 nM T35842 CKP26E 145976444 EC50 = 13 nM T35842 C7UJ8Q 145976863 EC50 = 57 nM T35842 CMS17N 145977650 EC50 = 13 nM T35842 CJ28PL 145980198 EC50 = 418 nM T35842 C0S1IN 145980719 IC50 = 50 nM T35842 CJ5T1Y 145987870 IC50 = 0.74 nM T35842 CF34MX 145988152 EC50 = 11 nM T35842 C39KYZ 145988867 EC50 = 25 nM T35842 C7WF3R 145989222 EC50 = 6.5 nM T35842 C50ZLS 145990599 EC50 = 10 nM T35842 CRSZ36 145993132 IC50 = 1.9 nM T35842 CDQZ25 145994283 IC50 = 80 nM T35842 C10FUX 145994325 IC50 > 5000 nM T35842 C5S4PT 24858479 EC50 > 1000 nM T35842 CHN0T4 24858480 EC50 = 76 nM T35842 CA83CB 24858481 EC50 = 810 nM T35842 CR08PO 24858629 IC50 > 1000 nM T35842 D00TSX 11672424 EC50 > 10000 nM T35842 D00VYC 44400370 Ki = 17.12 nM T35842 D01HTX 11707715 EC50 > 10000 nM T35842 D01VMU 44445082 IC50 > 10000 nM T35842 D02JVA 44408515 IC50 = 1500 nM T35842 D02MPZ 11535237 EC50 > 10000 nM T35842 D03AZC 25078192 Ki = 0.21 nM T35842 D04BOG 11629290 EC50 > 10000 nM T35842 D04YZZ 44445083 IC50 > 10000 nM T35842 D05LLI 11498895 EC50 > 1000 nM T35842 D05WNC 11520823 EC50 > 10000 nM T35842 D05XRI 44400401 Ki = 10.34 nM T35842 D06PNU 44409257 Ki = 2276 nM T35842 D06RTP 11700730 IC50 = 4000 nM T35842 D07DWH 44400402 Ki = 16.78 nM T35842 D07IBF 44400322 Ki > 500 nM T35842 D07SFD 44408443 IC50 = 1400 nM T35842 D07UXW 44408400 EC50 > 10000 nM T35842 D08DND 44445084 IC50 > 10000 nM T35842 D09LHF 44413535 EC50 = 77.4 nM T35842 D09OMI 44400400 Ki = 15.76 nM T35842 D09PDT 24774519 IC50 = 410 nM T35842 D09XCH 44400371 Ki = 147.07 nM T35842 D0A8ME 44400398 Ki = 67.09 nM T35842 D0B8GR 44413876 Ki = 13 nM T35842 D0B9NH 44408399 EC50 > 10000 nM T35842 D0C7VI 44400369 Ki = 0.57 nM T35842 D0F6GX 44409240 Ki = 4520 nM T35842 D0GN9K 24774602 IC50 = 412 nM T35842 D0L1MJ 11700739 IC50 = 3000 nM T35842 D0M2QK 44413536 EC50 = 67 nM T35842 D0M4EF 11593084 EC50 > 10000 nM T35842 D0N6AS 44158031 EC50 > 1000 nM T35842 D0N6KO 9938402 EC50 = 5 nM T35842 D0P4GI 11629326 EC50 > 10000 nM T35842 D0QW4A 24774356 IC50 > 10000 nM T35842 D0R0BY 44400320 Ki = 8.22 nM T35842 D0R5KO 44413537 EC50 = 1303.7 nM T35842 D0U1UZ 44413577 EC50 = 269.9 nM T35842 D0U5KM 11093672 EC50 = 4.3 nM T35842 D0U6XP 16724004 EC50 = 160 nM T35842 D0V5YV 44413592 EC50 = 5095.8 nM T35842 D0VD7R 44408408 EC50 > 10000 nM T35842 D0W1SM 44408413 EC50 = 1000 nM T35842 D0WG8P 44400321 Ki = 9.91 nM T35842 D0WI8M 44445085 IC50 = 2000 nM T35842 D0X1YL 25078242 Ki = 2.73 nM T35842 D0XQ5U 24774438 IC50 = 707 nM T35842 D0YB7F 92432 EC50 < 0.03162 nM T35842 D0ZD3M 44400399 Ki = 49.42 nM T30372 D01XBA 5035 IC50 = 33000 nM T30372 D02VMJ 50248 IC50 = 15000 nM T30372 D03RTS 2662 IC50 = 126000 nM T30372 D04AIT 5280445 IC50 = 27300 nM T30372 D07XGR 3339 IC50 = 61000 nM T30372 D08QIP 4887 IC50 = 7000 nM T30372 D09XZB 123631 IC50 = 148000 nM T30372 D0AZ3C 5291 IC50 = 297000 nM T30372 D0BP9C 193962 IC50 = 4000 nM T30372 D0N0TZ 60606 IC50 = 123000 nM T30372 D0Q3YO 1547484 IC50 = 124000 nM T30372 D0S5UH 2794 IC50 = 6000 nM T30372 D0J6AU 10152654 Ki = 125.89 nM T30372 D0L4FS 5280961 IC50 = 82700 nM T30372 D04YJU 9829836 IC50 = 12000 nM T30372 C5IF7O 2259 IC50 = 28000 nM T30372 C5Q6US 2540 IC50 = 42000 nM T30372 CY4WG9 3793 IC50 = 3000 nM T30372 C0OCW6 6240 IC50 = 189000 nM T30372 C4IU5T 6889 IC50 >> 10000 nM T30372 C53FYO 11840 IC50 >> 10000 nM T30372 CC1NT6 27990 IC50 = 98000 nM T30372 CJQ9A8 34200 IC50 >> 10000 nM T30372 CN8A2G 38296 IC50 >> 10000 nM T30372 CP8F7B 64143 IC50 = 144000 nM T30372 C0EH3Z 88695 IC50 >> 10000 nM T30372 CX82ZE 92303 IC50 = 129000 nM T30372 C0KV5M 236566 IC50 >> 10000 nM T30372 CTC3W8 370995 IC50 = 28000 nM T30372 C6B5KN 439487 IC50 = 3000 nM T30372 CF4V3X 441325 IC50 = 4000 nM T30372 CH2Y3N 441386 IC50 = 122000 nM T30372 C8UB5Z 654761 IC50 < 1000 nM T30372 C6EAL2 659466 IC50 < 600000 nM T30372 CMR0Q4 663743 IC50 < 1000 nM T30372 CNE93W 664316 IC50 = 73000 nM T30372 C5UXD8 665449 IC50 = 95000 nM T30372 CX06HK 701796 IC50 = 7000 nM T30372 C9TWY0 712283 IC50 = 70 nM T30372 C47PBN 715039 IC50 = 15000 nM T30372 C5BF4N 717599 IC50 = 30000 nM T30372 CGAR13 717866 IC50 = 30000 nM T30372 CK42MF 721475 IC50 = 10900 nM T30372 C0TFO9 724128 IC50 = 4100 nM T30372 CCP0J7 729558 IC50 = 90 nM T30372 CU4M6G 766854 IC50 = 50000 nM T30372 CE4L0Y 778602 IC50 = 710 nM T30372 C0GR6M 821625 IC50 > 120000 nM T30372 C1SEV9 833435 IC50 = 12000 nM T30372 C8YWA6 843629 IC50 = 1000 nM T30372 CF6KH2 870542 IC50 = 16000 nM T30372 CYKN64 873495 IC50 > 60000 nM T30372 CC2S1T 873501 IC50 > 120000 nM T30372 CM5TF1 898637 IC50 < 600000 nM T30372 COYG56 914535 IC50 = 890 nM T30372 CYZH47 963166 IC50 > 60000 nM T30372 C4LOG7 974754 IC50 = 106000 nM T30372 CAR76K 1088642 IC50 > 200000 nM T30372 CXZ2S1 1161245 IC50 = 12000 nM T30372 C3IT2O 1179204 IC50 = 30000 nM T30372 CRV8A9 1183113 IC50 = 800 nM T30372 CX4G5A 1246514 IC50 = 12000 nM T30372 CWD4U0 1305492 IC50 > 600000 nM T30372 C3UQ2C 1616653 IC50 = 700 nM T30372 C6H8JE 1633306 IC50 > 60000 nM T30372 C85YWF 1670121 IC50 > 200000 nM T30372 C67RBE 2013546 IC50 = 12000 nM T30372 CQK10R 2066617 IC50 = 3000 nM T30372 CC1A3F 2117743 IC50 = 30000 nM T30372 CA7DV8 2155684 IC50 = 30000 nM T30372 CH6NA7 2191015 IC50 < 1000 nM T30372 CV1Z9B 2235625 IC50 = 90000 nM T30372 CD3J6I 2263233 IC50 = 13200 nM T30372 CW6TN3 2327228 IC50 = 12000 nM T30372 CLR43Q 2341222 Ki = 32000 nM T30372 C7LC9N 2368254 IC50 = 30000 nM T30372 CG57WH 2382051 IC50 = 120000 nM T30372 CV6R1K 2514971 IC50 = 120000 nM T30372 C2R8NI 2726959 IC50 = 1200 nM T30372 CE8XK7 2768681 IC50 >> 10000 nM T30372 CC35FD 2808017 IC50 < 10000 nM T30372 CTK5Y8 2820493 IC50 = 3100 nM T30372 CL1K0J 2881154 IC50 > 60000 nM T30372 C5ZKX6 2998581 IC50 = 12000 nM T30372 CTO4G9 2998924 Ki = 6000 nM T30372 CBN01J 2999703 IC50 > 120000 nM T30372 CRNH81 3000182 IC50 = 38000 nM T30372 C98WUE 3239413 IC50 > 10000000 nM T30372 CV4JE8 3336226 IC50 = 12000 nM T30372 C0H5FK 3556842 Ki = 800 nM T30372 CQ0AR8 3704739 IC50 = 90000 nM T30372 CZG20R 3888858 IC50 = 3000 nM T30372 CT6ER0 3976161 IC50 = 1000 nM T30372 CER7Y3 4200465 IC50 = 12000 nM T30372 CQ3A6Z 4313265 IC50 = 500 nM T30372 C1JX2E 4403597 IC50 = 58000 nM T30372 C4G8FY 4437145 IC50 = 400 nM T30372 CLV48W 4438641 Ki = 70 nM T30372 C3DIU4 4474562 IC50 < 10000 nM T30372 CYXT47 4576615 IC50 = 1900 nM T30372 C45EIS 4592377 IC50 = 11000 nM T30372 C8WP3E 4650466 IC50 = 62000 nM T30372 CV8W5S 4798096 IC50 = 44000 nM T30372 C5B8AN 4828813 IC50 = 126000 nM T30372 C9ZIR2 4875671 IC50 = 18000 nM T30372 C8T3IE 5289424 Ki = 144.54 nM T30372 CIMS58 5308729 IC50 = 120000 nM T30372 C87WPI 5319895 IC50 = 9600 nM T30372 CHR31N 5346422 IC50 = 20000 nM T30372 C6HD5Z 5390849 IC50 = 1900 nM T30372 CUZN74 5412428 IC50 = 3800 nM T30372 CD39LW 5480198 IC50 > 20000 nM T30372 C03YRU 5495611 IC50 > 10000 nM T30372 C2DY4Q 5710398 IC50 = 1300 nM T30372 CJ2Q9I 6289371 IC50 > 17000 nM T30372 C0JDO7 6604839 IC50 = 158000 nM T30372 CV8XR4 6870649 IC50 > 10000 nM T30372 CAY81D 6875597 IC50 > 10000 nM T30372 CUWI14 6882251 IC50 > 10000 nM T30372 CQC06M 7149198 IC50 = 90000 nM T30372 CHO4P1 7224671 IC50 = 5000 nM T30372 CM9ZS4 7695054 IC50 = 1300 nM T30372 CCQG24 7700632 IC50 = 12000 nM T30372 CS69AZ 7728947 IC50 > 10000 nM T30372 C5DB4N 8893764 IC50 = 182000 nM T30372 CKJS68 9556622 IC50 > 10000 nM T30372 CHSM95 9563238 IC50 = 140 nM T30372 CW54YZ 9563572 IC50 > 10000 nM T30372 CI9BK1 9563573 IC50 = 300 nM T30372 CM0DB1 9569552 IC50 > 10000 nM T30372 C21FRT 9569914 IC50 = 10000 nM T30372 CJE6K7 9600754 IC50 > 10000 nM T30372 C3GZ4L 9601317 IC50 = 170 nM T30372 CNUV20 9616512 IC50 > 10000 nM T30372 CR97AP 9625075 IC50 > 10000 nM T30372 CM2A0J 9645531 IC50 = 320 nM T30372 CY6AE9 9651823 IC50 = 121000 nM T30372 CY05VN 9718959 IC50 > 10000 nM T30372 CTUS65 9726252 IC50 > 10000 nM T30372 CS2AZ9 9731214 IC50 > 10000 nM T30372 C79LKI 9737735 IC50 = 1300 nM T30372 C31TRH 9746003 IC50 > 10000 nM T30372 C30CBL 9753989 IC50 > 10000 nM T30372 CE42MQ 9809035 Ki = 0.9 nM T30372 CM9A4D 9878645 IC50 = 60 nM T30372 C0YMK4 9921964 IC50 = 40 nM T30372 C65WKU 9926053 IC50 = 41000 nM T30372 CEL43J 9965377 IC50 = 50 nM T30372 CP9US8 9970504 IC50 = 80 nM T30372 CO1JN6 9971885 IC50 = 80 nM T30372 CC05RX 9982218 IC50 > 120000 nM T30372 C1B5DC 10096920 IC50 = 10 nM T30372 CD6L1T 10098422 Ki = 16 nM T30372 CS82ZK 10107471 IC50 = 20 nM T30372 C34BJE 10331944 IC50 = 220 nM T30372 C72AYZ 10336662 IC50 = 60 nM T30372 CRD09K 10379340 IC50 = 70 nM T30372 CGN25S 10382804 IC50 = 20 nM T30372 CKCN24 10422411 IC50 = 230 nM T30372 C83HMU 10468445 IC50 = 200 nM T30372 C1LPY9 10468909 IC50 >> 10000 nM T30372 C47KUQ 10471660 IC50 = 2800 nM T30372 CJP85S 10642441 IC50 = 90000 nM T30372 CD8Q0U 10858632 IC50 > 10000 nM T30372 CYA40G 10859546 IC50 > 10000 nM T30372 C5PO2E 10860405 IC50 > 10000 nM T30372 CAD6T0 10864154 Ki = 54.6 nM T30372 C16MLB 10865176 Ki = 5 nM T30372 CM5J9L 10868441 IC50 > 10000 nM T30372 C5ZN1E 10870240 IC50 > 10000 nM T30372 C6F1AE 10870565 IC50 = 2800 nM T30372 CNC57A 10874460 Ki = 59.7 nM T30372 C6MB9W 10875534 Ki = 22.7 nM T30372 CW4CU5 10882968 IC50 > 10000 nM T30372 CF42QV 10883755 IC50 = 1000 nM T30372 CMO9Y1 10886114 Ki = 1.4 nM T30372 C0M5FA 10886544 Ki = 82.7 nM T30372 C3DBO6 10900297 IC50 > 10000 nM T30372 C9LWT7 10900890 IC50 > 10000 nM T30372 C1CI7A 10901721 IC50 = 3900 nM T30372 CA9ZC6 10907387 Ki = 2 nM T30372 C6HFQ9 10918624 Ki = 30.1 nM T30372 CGE8T6 10918632 Ki = 15 nM T30372 C1LPT2 10924138 IC50 > 10000 nM T30372 C9HML6 10934180 IC50 > 10000 nM T30372 CF3V0M 10934672 IC50 = 280 nM T30372 C3L5RH 10944513 IC50 = 270 nM T30372 CRUG35 10959957 IC50 = 1700 nM T30372 C6MH8B 10962390 Ki = 69.6 nM T30372 CJAO02 10972936 Ki = 7.8 nM T30372 CCFA87 10983274 IC50 = 300 nM T30372 CAU87Y 10989825 IC50 > 10000 nM T30372 CSO24N 11006217 Ki = 7.5 nM T30372 C1B8XK 11006491 Ki = 32.4 nM T30372 C32AOZ 11016982 Ki = 130.7 nM T30372 C56FMI 11027472 Ki = 1.3 nM T30372 CPUX50 11027483 Ki = 13.8 nM T30372 CD2O9P 11028084 Ki = 59.1 nM T30372 CL19TE 11028356 Ki = 2 nM T30372 CQ0I3S 11028538 Ki = 22 nM T30372 C5CLK8 11045180 IC50 > 10000 nM T30372 CJIS60 11049744 Ki = 5.8 nM T30372 CQXP76 11050104 Ki = 1.1 nM T30372 CZ9GD0 11055010 IC50 > 10000 nM T30372 C8ONW5 11059060 IC50 = 1600 nM T30372 C0OCV2 11064119 IC50 > 10000 nM T30372 CZIE19 11066029 IC50 > 10000 nM T30372 CUB45Z 11067581 IC50 = 7000 nM T30372 CYDC69 11068494 IC50 > 10000 nM T30372 CFT2K6 11068551 IC50 > 10000 nM T30372 CMP6K1 11071803 Ki = 1 nM T30372 C3IE6O 11075462 IC50 > 10000 nM T30372 CF94XH 11078891 IC50 > 10000 nM T30372 CC0Q9F 11081613 Ki = 4.8 nM T30372 CARU90 11082296 Ki = 31.2 nM T30372 CMYR45 11087445 IC50 > 10000 nM T30372 C0PYQ4 11100685 IC50 = 1400 nM T30372 CNO64I 11103527 Ki = 8 nM T30372 CC5AZ8 11103790 Ki = 216.3 nM T30372 CMC63T 11113842 Ki = 14.1 nM T30372 C7M4DW 11114280 Ki = 34.3 nM T30372 C5XD7Z 11114597 Ki = 10.4 nM T30372 CB0L4E 11117789 IC50 > 10000 nM T30372 CL1V8B 11124614 Ki = 44 nM T30372 CL68MX 11124691 Ki = 37 nM T30372 C3ED7J 11124720 Ki = 4.2 nM T30372 CSCK73 11140610 IC50 = 200 nM T30372 CV2ZY0 11145746 Ki = 4.6 nM T30372 CIV2E6 11161535 IC50 = 8000 nM T30372 CR8KV9 11161910 IC50 > 20000 nM T30372 C9ZNL4 11191320 Ki = 173 nM T30372 CNM0X6 11199052 IC50 = 5000 nM T30372 CW9G4R 11221479 IC50 = 5000 nM T30372 C1OQ8L 11266125 IC50 = 10000 nM T30372 C8NB1K 11266650 IC50 > 20000 nM T30372 CN2D7F 11278865 IC50 = 5000 nM T30372 CME0C5 11443502 Ki = 93.2 nM T30372 CB0G5Y 11594647 IC50 = 19 nM T30372 C5ZOM0 11656060 IC50 = 1.8 nM T30372 C5SZ9Q 11737693 IC50 > 20000 nM T30372 C8EZR3 11763189 Ki = 2.5 nM T30372 CSC7B5 11766901 Ki = 34.3 nM T30372 CGU6I7 11767007 Ki = 2.9 nM T30372 CJE2N6 11767014 Ki = 30.4 nM T30372 C3GHR0 11767148 Ki = 5.5 nM T30372 CF6O3X 11812006 IC50 > 10000 nM T30372 CC41US 11827588 Ki = 4.6 nM T30372 C5VJ2L 12007058 IC50 > 10000 nM T30372 C9WC6M 14655218 Ki = 501.19 nM T30372 CM2NQ4 15138473 IC50 > 17000 nM T30372 CTIE37 15308693 Ki = 6309.57 nM T30372 CR2GO6 15488850 Ki = 1584.89 nM T30372 CF0M4P 15488851 Ki = 7.943 nM T30372 C9LW6H 15985754 IC50 = 0.2 nM T30372 C8PL7J 16010307 IC50 = 12000 nM T30372 CYLP62 16043323 IC50 = 17 nM T30372 CY0FX8 16061496 IC50 = 210 nM T30372 CR36DE 17132316 IC50 = 9500 nM T30372 CGVS15 17414912 IC50 = 2700 nM T30372 CJU6A4 17421760 IC50 = 84000 nM T30372 C1EJ5S 17456138 IC50 = 3000 nM T30372 C2MDQ7 18143836 IC50 = 65100 nM T30372 CP2AX0 19171432 IC50 = 800 nM T30372 C9R1KG 20846819 IC50 = 12000 nM T30372 CCA21D 21008970 IC50 = 5200 nM T30372 C4MCB5 21008988 IC50 = 38400 nM T30372 CPN4C1 21235665 IC50 = 50000 nM T30372 C9ZQL7 23730357 IC50 > 50000 nM T30372 CRE7A4 23730473 IC50 > 50000 nM T30372 CK8XV4 24881399 IC50 = 370 nM T30372 C4OE1F 24881534 IC50 = 37 nM T30372 CZ21HD 24898027 Ki = 1.995 nM T30372 CQ1AF3 25032698 Ki = 250 nM T30372 C73KLE 25209862 IC50 = 0.26 nM T30372 CGV12I 25234547 IC50 = 80 nM T30372 CQNG94 25234548 IC50 = 800 nM T30372 CBD83K 25234550 IC50 > 3640 nM T30372 C26LYE 25234551 IC50 > 2000 nM T30372 CB51YF 25234552 IC50 = 110 nM T30372 CI16LB 25234553 IC50 = 1200 nM T30372 CBLN16 25234558 IC50 > 16000 nM T30372 CGD30O 25234561 IC50 = 820 nM T30372 CU38HV 25234562 IC50 > 20000 nM T30372 C2QP5B 25234577 IC50 > 33000 nM T30372 COB43C 25798545 IC50 >> 10000 nM T30372 CC2NR1 30209012 IC50 = 5300 nM T30372 CX9O4L 37020172 Ki = 82 nM T30372 CL96WQ 42633150 IC50 = 16 nM T30372 CZ5F4C 42633340 IC50 = 17 nM T30372 C5XV0H 42633341 IC50 = 1 nM T30372 CZS24P 42633520 IC50 = 0.2 nM T30372 CI78XT 42633521 IC50 = 0.4 nM T30372 CU6PL7 42633691 IC50 = 8 nM T30372 CQ9TR8 42633692 IC50 = 8 nM T30372 C6FJW2 42634249 IC50 = 3 nM T30372 C9EN0G 42634411 IC50 = 3 nM T30372 C2ZXJ7 42634578 IC50 = 2 nM T30372 CI25RJ 42634754 IC50 = 8 nM T30372 CZ6B1F 42635119 IC50 = 0.2 nM T30372 C5X4WG 42635483 IC50 = 6 nM T30372 CJ3Y2H 42641702 Ki = 1040 nM T30372 C3K0GH 42641703 Ki = 6760 nM T30372 C89JXT 42641704 Ki = 940 nM T30372 CE8U0Z 42641705 Ki = 100 nM T30372 CAP95J 42641817 Ki = 130 nM T30372 C9H1VW 42641818 Ki = 350 nM T30372 CFA3V2 42641819 IC50 = 27 nM T30372 C2X8UR 42641820 Ki = 1220 nM T30372 CFE71S 43091000 Ki = 12100 nM T30372 CP0Q4T 44142116 IC50 = 1 nM T30372 CBF74T 44142124 IC50 = 0.3 nM T30372 C25ELB 44143088 IC50 = 0.2 nM T30372 CL0M7R 44143089 IC50 = 13 nM T30372 CXGF58 44143090 IC50 = 0.4 nM T30372 C9QDC0 44143091 IC50 = 251 nM T30372 CGWH04 44234900 IC50 = 25000 nM T30372 CEQ28K 44234901 IC50 = 14000 nM T30372 C0NRK9 44234902 IC50 = 3000 nM T30372 C1QT6M 44234903 IC50 = 2000 nM T30372 CMA0X2 44234904 IC50 = 7000 nM T30372 C0A3SI 44234905 IC50 = 8000 nM T30372 C5L2QT 44235158 IC50 > 100000 nM T30372 CI7M1X 44235159 IC50 > 100000 nM T30372 CKP9S1 44235160 IC50 = 200 nM T30372 CNWO25 44235161 IC50 = 1000 nM T30372 C0HI4W 44235162 IC50 = 2000 nM T30372 CSJ56Q 44235163 IC50 > 100000 nM T30372 C8BHS0 44235164 IC50 = 6000 nM T30372 C9WLK1 44235396 IC50 = 8000 nM T30372 C48HIS 44235398 IC50 = 500 nM T30372 C7I2GO 44235399 IC50 = 800 nM T30372 CN21AC 44235400 IC50 = 11000 nM T30372 CI7FR4 44324369 IC50 > 10000 nM T30372 C3L8JZ 44324425 IC50 > 10000 nM T30372 C9EOY5 44324553 IC50 = 2800 nM T30372 CAF72Y 44327540 IC50 > 1000 nM T30372 CJ5W0G 44332538 Ki = 384 nM T30372 C1KD2V 44332539 Ki = 983 nM T30372 C7XQY2 44332540 Ki = 53 nM T30372 C2FHG7 44332555 Ki = 202 nM T30372 C6QOU0 44332714 Ki = 366 nM T30372 C83QDU 44332915 Ki = 274 nM T30372 CKO7M9 44338665 IC50 = 5000 nM T30372 CMDG36 44344692 IC50 >> 10000 nM T30372 CK14BJ 44344949 IC50 >> 10000 nM T30372 CN2HW5 44344950 IC50 = 80000 nM T30372 C4B5LJ 44344990 IC50 >> 10000 nM T30372 CLG09E 44391871 IC50 = 40 nM T30372 C3LV8U 44391872 IC50 = 30 nM T30372 C5BW3L 44391882 IC50 = 30 nM T30372 C01MLD 44391883 IC50 = 40 nM T30372 C8F3WR 44391899 IC50 > 10000 nM T30372 CZ63QT 44391902 IC50 = 3000 nM T30372 C5QR1V 44391906 IC50 = 30 nM T30372 C3T8YW 44391915 IC50 = 80 nM T30372 CKC4P5 44411027 Ki = 900 nM T30372 C2MDN7 44411237 Ki = 790 nM T30372 CGQ6I3 44414939 IC50 > 20000 nM T30372 CSB61N 44414940 IC50 > 5000 nM T30372 C5ZXF6 44414941 IC50 > 7000 nM T30372 CU2CN4 44443885 IC50 = 20 nM T30372 C10MUK 44443886 IC50 = 50 nM T30372 CS7TI4 44446955 Ki = 3300 nM T30372 CB96GK 44446958 Ki = 170 nM T30372 CW0MP5 44446964 Ki = 3600 nM T30372 CNZ2U6 44446971 Ki = 980 nM T30372 C3G7JF 44446973 Ki = 97 nM T30372 CQ59ST 44446977 Ki = 80 nM T30372 CZX0L4 44446981 Ki = 50 nM T30372 CZ3HK1 44446983 Ki = 92 nM T30372 CRH4Q0 44446985 Ki = 280 nM T30372 CIYS47 44446987 Ki = 71 nM T30372 C4VRK2 44446989 Ki = 150 nM T30372 CIR4P7 44446992 Ki = 350 nM T30372 CCR83O 44446993 Ki = 45 nM T30372 CDG1V2 44446994 Ki = 1700 nM T30372 C1H0KV 44446996 Ki = 19 nM T30372 C8DN1C 44450464 IC50 = 95000 nM T30372 CV2U4O 44450928 Ki = 4.365 nM T30372 CF4Z9G 44450953 Ki > 10000 nM T30372 C6ZFL9 44450954 Ki > 5011.87 nM T30372 C5LT9B 44450978 Ki > 10000 nM T30372 COY83D 44459953 IC50 = 1260 nM T30372 CV05NU 44459954 IC50 = 790 nM T30372 CP70SN 44459955 IC50 = 1580 nM T30372 CP6K5L 44459956 IC50 = 890 nM T30372 C8K5EZ 44459957 IC50 = 890 nM T30372 C0VX8S 44459958 IC50 = 890 nM T30372 C8INY0 44459961 IC50 = 710 nM T30372 C6OJ9P 44459963 IC50 = 890 nM T30372 CK1S6Q 44459964 IC50 = 1410 nM T30372 C1HPA9 44459965 IC50 = 79 nM T30372 CRX1S4 44459966 IC50 = 30 nM T30372 C8Z4WO 44459967 IC50 = 2 nM T30372 C73YVF 44459971 IC50 = 126 nM T30372 C21WFB 44459973 IC50 = 40 nM T30372 CS49LV 44459975 IC50 = 2 nM T30372 CTA1L6 44459976 IC50 = 60 nM T30372 C86ORE 44459987 IC50 = 4 nM T30372 CC1GE2 44459988 IC50 = 10 nM T30372 C15QAC 44459990 IC50 = 2239 nM T30372 CY6J1H 44459993 IC50 = 63 nM T30372 CX1JS8 44460078 IC50 = 18 nM T30372 CSXN79 44460079 IC50 = 316 nM T30372 C57JYH 44460080 IC50 = 63 nM T30372 C4N3ED 44460081 IC50 = 71 nM T30372 CT54YR 44460082 IC50 = 50 nM T30372 CP35KH 44560381 IC50 > 100000 nM T30372 C94XLJ 44560432 IC50 = 43000 nM T30372 CQMP31 44560527 IC50 = 32000 nM T30372 CJ49RU 44563607 IC50 > 10000 nM T30372 CBC7F5 44563608 IC50 = 2000 nM T30372 C2WU1D 45104217 Ki = 190 nM T30372 CQ2M6K 45267066 IC50 = 4000 nM T30372 CQ54ZI 45267072 IC50 = 23000 nM T30372 CZA37T 45267075 IC50 = 17000 nM T30372 CM4CA2 45267082 IC50 > 100000 nM T30372 CL7E2O 45267085 IC50 > 100000 nM T30372 C0EBT2 45267928 IC50 = 6000 nM T30372 CR9CL5 45267936 IC50 = 33000 nM T30372 C9ZT5O 45267942 IC50 = 62000 nM T30372 CN8E6P 45268807 IC50 = 7000 nM T30372 CD9NE5 45268812 IC50 = 14000 nM T30372 CS0G9U 45268823 IC50 = 83000 nM T30372 CF79AK 45268824 IC50 > 100000 nM T30372 CH47PV 45268826 IC50 > 100000 nM T30372 CVQ0Y8 45269656 IC50 = 36000 nM T30372 CWL1S7 45270483 IC50 = 2000 nM T30372 C4EG2P 45270486 IC50 = 6000 nM T30372 CDZS86 45270498 IC50 = 32000 nM T30372 CJ7K6C 45270499 IC50 = 36000 nM T30372 CA4LK0 45270500 IC50 = 52000 nM T30372 C0T3UQ 45270502 IC50 > 100000 nM T30372 CDJ6M1 45271310 IC50 = 3000 nM T30372 C2VQF0 45271317 IC50 = 10000 nM T30372 C9EZ0O 45271319 IC50 = 41000 nM T30372 C6W2TQ 45271327 IC50 = 42000 nM T30372 CKX9A8 45271333 IC50 = 17000 nM T30372 C5BV4D 45272205 IC50 = 6000 nM T30372 CR7ZL8 45272209 IC50 = 11000 nM T30372 CQT96I 45272210 IC50 = 8000 nM T30372 CR82TE 45272214 IC50 = 18000 nM T30372 CY06MN 45272218 IC50 = 38000 nM T30372 CP4CH7 45273055 IC50 > 100000 nM T30372 CUR43K 45273062 IC50 = 17000 nM T30372 C4WCZ2 45273074 IC50 > 100000 nM T30372 CO74ZC 45485239 IC50 = 12000 nM T30372 CT9UF1 45485251 IC50 = 12000 nM T30372 C26UHC 45485273 IC50 = 60000 nM T30372 C9TJG5 46175111 IC50 = 50 nM T30372 C38HWY 46878211 Ki = 600 nM T30372 CZ43KH 46878212 Ki = 2500 nM T30372 C98HGD 46882170 IC50 = 10000 nM T30372 CFW1K3 46882171 IC50 = 2000 nM T30372 CO5B7D 46882172 IC50 = 1000 nM T30372 CV4H0Q 46882173 IC50 = 2000 nM T30372 CQDL61 46882211 IC50 = 5000 nM T30372 CI72MY 46882212 IC50 = 1000 nM T30372 CA4XR8 46882213 IC50 = 6000 nM T30372 CG53ZX 46882251 IC50 > 100000 nM T30372 CWBM02 46898369 IC50 = 86000 nM T30372 CFOZ79 46899194 IC50 = 81000 nM T30372 CJUA90 49799570 IC50 = 700 nM T30372 C4VLK6 49837085 IC50 > 500000 nM T30372 CBM27Y 49837191 IC50 > 500000 nM T30372 CG08WO 49853260 IC50 = 77500 nM T30372 C4I0JY 50925524 IC50 = 0.1 nM T30372 C7DO0F 52941283 IC50 = 7 nM T30372 CU1TW6 52941414 IC50 = 7 nM T30372 C9MK7J 52942931 IC50 = 183 nM T30372 C4TY6S 52943722 IC50 = 380 nM T30372 CQ6N0I 52943841 IC50 > 10000 nM T30372 CV8L9Z 52945985 IC50 = 33 nM T30372 CLJ83U 52946267 IC50 = 510 nM T30372 CT28XU 52947761 IC50 = 130 nM T30372 CI02EQ 56643423 IC50 = 24000 nM T30372 CLW0X8 57398579 IC50 = 180000 nM T30372 COYW71 58336677 Ki = 10 nM T30372 CN01HD 60639592 Ki = 142 nM T30372 CZ6FH9 67298247 Ki = 39.81 nM T30372 CJOF37 67298501 Ki = 7.943 nM T30372 C2UN6D 71452029 IC50 = 10200 nM T30372 CG8T7Z 71452030 IC50 = 9500 nM T30372 C78BKL 71455561 IC50 = 6600 nM T30372 CS4M7Q 71456690 IC50 = 30 nM T30372 CZT23D 71459213 IC50 = 7000 nM T30372 CAI9X6 71460991 IC50 = 10800 nM T30372 CKLC20 71460992 IC50 = 11800 nM T30372 CXEF28 71462724 IC50 = 8700 nM T30372 C5GB6C 71540695 IC50 = 300 nM T30372 C54CNP 73345966 IC50 = 3000 nM T30372 C5QX3P 73352106 IC50 < 10000 nM T30372 CGFY52 73353564 IC50 = 6900 nM T30372 CW9NU4 73895627 Ki = 17 nM T30372 CHX9B4 90481669 IC50 = 40 nM T30372 CM9WE5 90481670 IC50 = 400 nM T30372 CPA9Y1 90486834 IC50 = 400 nM T30372 CZG92D 90644871 IC50 = 11200 nM T30372 CNE83B 90655102 IC50 = 1600 nM T30372 CF5Y1M 90655103 IC50 = 13500 nM T30372 CS8FZ9 90655104 IC50 = 12700 nM T30372 C1MP6L 90655105 IC50 = 8200 nM T30372 CC19XE 90655106 IC50 = 23900 nM T30372 C3SQ7W 90655107 IC50 = 9900 nM T30372 C4FSI3 90655108 IC50 = 600 nM T30372 CAY38G 90655109 IC50 = 540 nM T30372 C2NY0I 90655110 IC50 = 620 nM T30372 CIS56R 90663177 Ki = 220 nM T30372 CU71EO 90663180 Ki = 360 nM T30372 CX37IK 90663181 Ki = 48 nM T30372 C73TBD 90668194 Ki = 29.7 nM T30372 C2PAK4 90668198 Ki = 13.3 nM T30372 CO1VD9 90668199 Ki = 3.7 nM T30372 CK0AF8 101889645 IC50 = 21600 nM T30372 C7I4XF 101889646 IC50 = 8700 nM T30372 C56VIF 118712447 IC50 = 4800 nM T30372 C4UJ7G 118712449 IC50 = 10 nM T30372 C5ALU2 118719334 IC50 = 12000 nM T30372 CMBG29 118724585 IC50 = 7100 nM T30372 C5D6MO 122189123 IC50 = 600 nM T30372 C05AYZ 122189136 IC50 = 400 nM T30372 CRAT04 122189137 IC50 = 70 nM T30372 CH9Z4P 122189142 IC50 = 8 nM T30372 CJ04AZ 122193587 IC50 = 1350 nM T30372 CC6K9M 122193588 IC50 = 560 nM T30372 C10NKI 122193589 IC50 = 340 nM T30372 C2B3OY 122193866 IC50 = 1100 nM T30372 CLO27Y 122193867 IC50 = 23000 nM T30372 CT6H1N 122193868 IC50 = 3590 nM T30372 CPJ42N 122193869 IC50 = 125 nM T30372 C9QOP2 122193870 IC50 = 63 nM T30372 C1G3SI 122193871 IC50 = 5 nM T30372 CK8LM4 122193872 IC50 = 25 nM T30372 C2E6DP 122193873 IC50 = 124 nM T30372 C3X5SE 122193874 IC50 = 880 nM T30372 CHWC98 122193875 IC50 = 790 nM T30372 C6CN5X 122193876 IC50 = 75 nM T30372 CNJ3F4 122193877 IC50 = 3 nM T30372 C1ZO2L 122193878 IC50 = 467 nM T30372 C4QX5O 122193879 IC50 = 2820 nM T30372 CJ4KX8 127030097 IC50 = 3300 nM T30372 CPE2H1 127031325 IC50 = 600 nM T30372 CEF0V2 127033016 IC50 = 19000 nM T30372 CTO0G7 127045313 IC50 = 111000 nM T30372 CI9K6W 127045316 IC50 = 2400 nM T30372 C8Q7WR 127045466 IC50 = 85000 nM T30372 C0U6GR 134134734 Ki = 130 nM T30372 CD5NI4 134134799 Ki = 0.44 nM T30372 CW3B7G 134137121 Ki = 28 nM T30372 C4CT5Z 134139989 Ki = 25 nM T30372 C4HN8V 134148867 Ki = 16 nM T30372 CH98KJ 134154138 Ki = 11 nM T30372 C2UMT4 134157443 Ki = 130 nM T30372 CQV56G 135401155 IC50 = 600 nM T30372 C3QBE6 135419539 IC50 > 100000 nM T30372 CGV4W2 135439445 IC50 = 21000 nM T30372 CYV68B 135860621 IC50 = 23000 nM T30372 CPJ4N6 135860627 IC50 = 12000 nM T30372 CUCA37 135869166 IC50 > 100000 nM T30372 CGO97R 136029168 IC50 = 3000 nM T30372 CRS8X2 136035726 IC50 = 20400 nM T30372 CB08OL 136035727 IC50 = 400 nM T30372 CJY03Z 136044099 IC50 = 15100 nM T30372 CIC5F3 136099759 IC50 > 100000 nM T30372 CWH9T0 136099760 IC50 = 78000 nM T30372 CPZ45M 136116847 IC50 = 44700 nM T30372 CBY17U 136229787 IC50 = 40 nM T30372 CF8RV6 136229788 IC50 = 200 nM T30372 CVHU35 136229843 IC50 = 52200 nM T30372 CGS41D 136242670 IC50 = 74800 nM T30372 CXT0S9 136242672 IC50 = 45900 nM T30372 CK5Z4N 136242673 IC50 = 83900 nM T30372 CK14RX 145961420 IC50 = 9000 nM T30372 CEHT46 145963780 Ki = 398107.17 nM T30372 CWHR24 145963809 Ki = 25118.86 nM T30372 CG4V3W 145963956 Ki = 3981.07 nM T30372 CRU9S4 145964832 Ki = 1.585 nM T30372 CV43LX 145965335 Ki = 125892.54 nM T30372 C6MK4H 145965352 Ki = 100 nM T30372 CT17MJ 145967290 Ki = 10000 nM T30372 CGUS39 145968211 Ki = 199526.23 nM T30372 CI43YB 145973712 Ki = 6309.57 nM T30372 C2I0BM 145974244 Ki = 1.585 nM T30372 CNC48W 145982661 IC50 = 340 nM T30372 CMS4E9 145982820 IC50 = 80 nM T30372 CU5Z9F 145983387 IC50 = 3750 nM T30372 C1OEA0 145983615 IC50 = 630 nM T30372 C3LH7B 145984676 IC50 = 20 nM T30372 CJK42D 145985003 IC50 = 300 nM T30372 C8AM0K 145985030 IC50 > 2000 nM T30372 CURI53 145985037 IC50 = 20 nM T30372 CHCP90 145985556 IC50 = 330 nM T30372 CBK3G5 145985888 IC50 = 200 nM T30372 C50ERM 145986467 Ki = 5500 nM T30372 C85RXZ 145987523 Ki = 30900 nM T30372 C8NW1T 145990306 Ki = 1800 nM T30372 C70GTM 145990424 Ki = 7700 nM T30372 CQR52M 145990979 Ki = 7600 nM T30372 CH7WO9 145994261 Ki = 710 nM T30372 CJ2DW5 155510635 Ki = 79.43 nM T30372 CKT12D 155510715 Ki = 123 nM T30372 CW2VG7 155513724 Ki = 34.62 nM T30372 C31OBN 155513845 Ki = 168.02 nM T30372 CF01VN 155514418 Ki = 398.11 nM T30372 CX0ZB9 155514813 Ki = 360.08 nM T30372 C9NG5J 155514973 IC50 = 235000 nM T30372 C27SKJ 155515029 IC50 = 1.08 nM T30372 C8HP4U 155515082 Ki > 10000 nM T30372 C9VSY4 155515758 Ki = 37000 nM T30372 CJ6Z4N 155515766 Ki = 50.12 nM T30372 C5U6FM 155517896 IC50 = 0.73 nM T30372 CYL03V 155518363 Ki = 1995.26 nM T30372 CYL43J 155518582 Ki = 1140 nM T30372 CKJ9V2 155519071 IC50 = 0.25 nM T30372 CTO3W8 155519600 Ki = 141.72 nM T30372 CH62WS 155521212 Ki = 4000 nM T30372 COIR58 155522309 Ki = 2200 nM T30372 C0EWD4 155522491 Ki = 1.585 nM T30372 C85PHT 155522699 Ki > 10000 nM T30372 CO2Y0C 155523098 Ki = 280 nM T30372 C3OC1G 155523633 Ki = 5500 nM T30372 C6M1FK 155524435 Ki = 3981.07 nM T30372 CC9X2D 155525224 Ki = 398.11 nM T30372 CD7WG5 155525553 IC50 = 2.89 nM T30372 CDB4X8 155525667 Ki = 940 nM T30372 C6ZS1U 155529120 Ki = 3400 nM T30372 C87DAI 155530185 Ki = 316.23 nM T30372 CAK7H1 155532577 Ki = 38.78 nM T30372 CO50BS 155532888 Ki = 3000 nM T30372 C0WZD4 155533248 IC50 = 81 nM T30372 C5LHT6 155533365 Ki = 870 nM T30372 CF7Y6A 155534455 IC50 = 8100 nM T30372 C92YHN 155535180 IC50 = 1.35 nM T30372 CUW76I 155535429 Ki = 142.99 nM T30372 CIQ84V 155535610 Ki = 30048.4 nM T30372 CZ5X9D 155536101 Ki = 3.6 nM T30372 CZ59GS 155536157 Ki = 1.585 nM T30372 CB4MT7 155537119 IC50 = 1.07 nM T30372 CNMR90 155537964 IC50 = 1.2 nM T30372 CYB7N2 155538310 Ki = 570 nM T30372 C83AUP 155538690 Ki > 35000 nM T30372 C5Q8YO 155539200 Ki = 745.68 nM T30372 CXHT61 155539577 IC50 = 37.14 nM T30372 CTV4B7 155539870 IC50 = 0.49 nM T30372 CFRP81 155539888 Ki > 10000 nM T30372 CO3ZF7 155541809 Ki = 88 nM T30372 C2X0YP 155541949 Ki = 870 nM T30372 C2Q1RP 155543092 Ki = 4.009 nM T30372 CSPL93 155544114 Ki = 1420 nM T30372 C43ZKT 155544277 IC50 = 0.84 nM T30372 CB94ZI 155544429 IC50 = 1.15 nM T30372 CIZ8A6 155544625 IC50 = 0.47 nM T30372 CQW2L9 155545346 Ki = 0.631 nM T30372 C8Y4UM 155546877 IC50 = 537000 nM T30372 CFN30H 155547862 Ki > 5000 nM T30372 CY2TK7 155547967 Ki > 10000 nM T30372 C6ER3C 155550821 Ki = 1710 nM T30372 C3TS9N 155552318 Ki = 1000 nM T30372 CCF86H 155553085 Ki = 280 nM T30372 C8Z7GU 155553621 Ki = 63.1 nM T30372 C3OX6R 155554092 Ki = 4061.31 nM T30372 C2P9GA 155554760 IC50 = 0.8 nM T30372 CR0LC5 155555416 Ki = 25000 nM T30372 CWD8H4 155556369 Ki = 3400 nM T30372 C6O9FK 155556968 Ki = 280 nM T30372 C2AIC6 155559777 IC50 = 0.76 nM T30372 C15VEM 155561956 Ki = 405.84 nM T30372 CRO9V2 155561992 IC50 = 3.69 nM T30372 CV2N1W 155565585 Ki = 2511.89 nM T30372 C1N3AJ 155565629 Ki = 50.12 nM T30372 CW30IO 155567009 Ki = 2511.89 nM T30372 CVYI25 155567173 Ki = 4800 nM T30372 C6XG1Q 155568133 Ki = 710 nM T30372 C4ABY3 155568252 Ki = 251.19 nM T30372 C87EYK 155568784 Ki = 370 nM T30372 C63ZMF 4388929 IC50 = 17000 nM T30372 CK23AB 44450298 IC50 = 45000 nM T30372 CS2KV7 91935567 IC50 = 68000 nM T30372 CFA2Z8 91935568 IC50 = 100000 nM T30372 C3ULB9 91935569 IC50 = 73000 nM T30372 D01BQI 25798544 IC50 = 2000 nM T30372 D01HRG 12884 IC50 >> 10000 nM T30372 D02GOH 6604822 IC50 = 30000 nM T30372 D03JDL 135665263 IC50 > 60000 nM T30372 D03TPH 87203 IC50 >> 10000 nM T30372 D04FMU 625239 IC50 = 12000 nM T30372 D05CCT 4139 IC50 = 85000 nM T30372 D05VOH 5282367 IC50 = 18000 nM T30372 D06DKB 661700 Ki = 2000 nM T30372 D07NVK 25234549 IC50 = 860 nM T30372 D07PZF 16061497 IC50 = 24 nM T30372 D07XQR 1010578 IC50 = 12000 nM T30372 D08DEG 598633 IC50 = 12000 nM T30372 D08NYF 6870109 IC50 = 280 nM T30372 D08TMM 9851116 IC50 = 4 nM T30372 D09BXH 8147464 IC50 = 87000 nM T30372 D09FGQ 123985 IC50 = 400 nM T30372 D0A1CM 5281855 IC50 = 220000 nM T30372 D0DT5K 6875577 IC50 = 560 nM T30372 D0G2DQ 4669250 IC50 >> 10000 nM T30372 D0GP7D 54686376 IC50 = 95000 nM T30372 D0J3HR 10899142 IC50 = 1360 nM T30372 D0L7GI 2877914 IC50 = 12000 nM T30372 D0MF5Y 5281614 IC50 = 30000 nM T30372 D0N2QX 9580972 IC50 = 480 nM T30372 D0O0LU 264734 IC50 >> 10000 nM T30372 D0O5TA 2175573 IC50 = 6000 nM T30372 D0S2IS 10356636 IC50 = 310 nM T30372 D0S2NU 5363470 IC50 = 560 nM T30372 D0SP2O 7054 IC50 >> 10000 nM T30372 D0TZ5V 690109 IC50 = 3500 nM T30372 D0U3JD 16358 IC50 >> 10000 nM T30372 D0UL6C 7695053 IC50 = 460 nM T30372 D0V8DQ 9583002 IC50 = 50 nM T30372 D0W1AW 4234241 IC50 = 15000 nM T30372 D0ZR2T 2732752 IC50 >> 10000 nM T63966 D01PZD 5329098 IC50 = 8 nM T63966 D01ZRI 6450551 IC50 = 0.1 nM T63966 D03ZBT 11626560 IC50 > 1000 nM T63966 D07POC 176870 IC50 > 1000 nM T63966 D09GDD 11167602 IC50 = 1.5 nM T63966 D0G6QF 3081361 IC50 = 100 nM T63966 D0H0EQ 24826799 IC50 = 20.9 nM T63966 D0IQ6P 25102847 IC50 = 12 nM T63966 D0R0FO 9823820 IC50 = 22 nM T63966 D0R0MW 5329102 IC50 = 1 nM T63966 D0W5HK 216239 IC50 = 18 nM T63966 D00DRL 44137946 IC50 = 10 nM T63966 D02UFQ 11620908 IC50 > 10000 nM T63966 D02WVT 25031915 IC50 = 7 nM T63966 D03LWG 53235510 IC50 = 1510 nM T63966 D03QLG 9917013 IC50 = 209 nM T63966 D05PZB 135398495 IC50 = 10 nM T63966 D07HRU 9549295 IC50 = 1 nM T63966 D07KYT 24889392 IC50 > 10000 nM T63966 D07PNT 10433653 IC50 = 20 nM T63966 D08HOM 46207586 IC50 = 32 nM T63966 D09VMI 9933475 IC50 = 5 nM T63966 D0A1AQ 5329099 IC50 = 28 nM T63966 D0A1WN 11714580 IC50 = 890 nM T63966 D0D1GF 42642645 IC50 = 0.8 nM T63966 D0E3TC 44259 IC50 = 8.19 nM T63966 D0FD6D 11751922 IC50 = 3 nM T63966 D0G2QH 10297043 IC50 = 59 nM T63966 D0HS5V 11234052 Ki = 60 nM T63966 D0IQ0Z 46885626 IC50 = 42 nM T63966 D0M0XB 10302451 IC50 > 100000 nM T63966 D0M9QZ 11485656 IC50 = 37 nM T63966 D0P6DJ 151194 IC50 = 54 nM T63966 D0T2ER 24767976 IC50 = 3.2 nM T63966 D0W7JZ 9911830 IC50 = 0.21 nM T63966 D03BNU 59604787 IC50 > 3500 nM T63966 D0YK9D 9956119 IC50 > 5000 nM T63966 D00DQX 11667893 IC50 = 2 nM T63966 D0H4GI 10275001 IC50 = 16 nM T63966 D0L5YF 5329032 IC50 = 700 nM T63966 D0T3ME 156422 IC50 = 250 nM T63966 C6Y9CV 151193 IC50 = 110 nM T63966 CK0L4O 442514 IC50 = 2900 nM T63966 C4MNG8 445840 IC50 = 2800 nM T63966 COB86I 1474850 IC50 = 22000 nM T63966 C2GSN6 1475052 IC50 = 11000 nM T63966 CFVK40 3008950 IC50 = 19200 nM T63966 CD8UW1 3008956 IC50 > 50000 nM T63966 CCD93P 3008957 IC50 = 15200 nM T63966 CU64VM 3008958 IC50 > 50000 nM T63966 C8F0KM 3008959 IC50 = 26800 nM T63966 CV8R9Z 3008960 IC50 > 50000 nM T63966 C8EZ6O 3008961 IC50 > 50000 nM T63966 CX95SU 3008962 IC50 = 45900 nM T63966 C9B2MN 3008963 IC50 = 42700 nM T63966 C9E7BW 3008964 IC50 > 50000 nM T63966 CGK91Q 3008965 IC50 > 50000 nM T63966 CB3G6R 4913175 IC50 = 300 nM T63966 CH1G9Q 5147149 IC50 = 170 nM T63966 C0RXL8 5326956 IC50 = 15.49 nM T63966 CQL3C9 5329005 IC50 = 26000 nM T63966 C9OQZ0 5329007 IC50 = 800 nM T63966 C2S5DQ 5329008 IC50 > 33000 nM T63966 CFW19M 5329009 IC50 > 100000 nM T63966 C2FO4B 5329010 IC50 = 30 nM T63966 CZU0K3 5329011 IC50 = 400 nM T63966 C21WXV 5329012 IC50 = 30 nM T63966 CJ68OQ 5329013 IC50 < 2 nM T63966 CEJR83 5329014 IC50 = 900 nM T63966 COS5M9 5329015 IC50 = 1500 nM T63966 CKFS07 5329016 IC50 = 3 nM T63966 CC1EO4 5329017 IC50 = 300 nM T63966 CGC01T 5329018 IC50 = 300 nM T63966 C1XJL0 5329019 IC50 = 1100 nM T63966 C9SZ4Q 5329020 IC50 = 200 nM T63966 C5DO1Y 5329021 IC50 = 300 nM T63966 C2YDI8 5329022 IC50 = 500 nM T63966 CW3OV5 5329023 IC50 = 800 nM T63966 C6HSX8 5329024 IC50 = 1200 nM T63966 CP37NS 5329025 IC50 = 100 nM T63966 C3VHF6 5329026 IC50 = 100 nM T63966 CSRF48 5329027 IC50 = 500 nM T63966 CB6V5Y 5329028 IC50 = 300 nM T63966 C6AN1O 5329029 IC50 > 100000 nM T63966 C04EAP 5329030 IC50 = 1500 nM T63966 C1Y5QP 5329031 IC50 = 300 nM T63966 C4VLR8 5329033 IC50 = 800 nM T63966 CLT7J9 5329034 IC50 = 8100 nM T63966 C9VX8C 5329040 IC50 = 3900 nM T63966 CK6T4U 5329042 IC50 = 500 nM T63966 CA81XO 5329045 IC50 = 300 nM T63966 C4T3MO 5329046 IC50 = 500 nM T63966 CQ15KR 5329049 IC50 = 700 nM T63966 C49KNS 5329050 IC50 = 450 nM T63966 C3C1EZ 5329051 IC50 = 800 nM T63966 C0H5XL 5329052 IC50 = 500 nM T63966 CW0KA8 5329053 IC50 = 150 nM T63966 COEN93 5329054 IC50 = 200 nM T63966 CATX52 5329055 IC50 = 700 nM T63966 CEQP41 5329056 IC50 = 500 nM T63966 CDV4C9 5329057 IC50 = 500 nM T63966 C4RUV5 5329453 IC50 = 210 nM T63966 C5RK3H 5330188 IC50 > 100000 nM T63966 CD7U5B 5330196 IC50 > 100000 nM T63966 CB23PA 5330197 IC50 > 100000 nM T63966 C2DCW3 5916724 IC50 = 30000 nM T63966 CV2KQ1 6326407 IC50 = 50 nM T63966 CF46XV 6326408 IC50 = 63000 nM T63966 C2H3UZ 6326413 IC50 = 2300 nM T63966 C49DUV 6326414 IC50 = 60 nM T63966 C7ZB6K 6326415 IC50 = 70 nM T63966 CJN34Y 6326416 IC50 = 9800 nM T63966 C9WDE8 6326417 IC50 > 10000 nM T63966 C1P5HD 6326418 IC50 = 760 nM T63966 CDWI70 6326419 IC50 = 620 nM T63966 CZJ1R9 6326420 IC50 > 10000 nM T63966 CPO78D 6326421 IC50 = 2600 nM T63966 CBD49X 6326422 IC50 = 420 nM T63966 C53UGK 6419378 IC50 = 650 nM T63966 CK3A1M 6419379 IC50 = 3000 nM T63966 C1Y8LP 6419380 IC50 = 1700 nM T63966 C3DO7L 6419381 IC50 = 470 nM T63966 CJ6QB4 6419382 IC50 = 230 nM T63966 CQO68G 6419383 IC50 = 240 nM T63966 CV5C7R 6419384 IC50 = 3600 nM T63966 C27ZIA 6419385 IC50 = 260 nM T63966 C6L5HS 6419386 IC50 = 60 nM T63966 C3CQW0 6419387 IC50 = 40 nM T63966 CWOA63 6419388 IC50 = 240 nM T63966 CZVU64 6419389 IC50 = 230 nM T63966 C9FN4B 6419390 IC50 = 330 nM T63966 CN53YW 6419391 IC50 = 80 nM T63966 C17NWJ 6419392 IC50 = 70 nM T63966 C13IRC 6419393 IC50 = 260 nM T63966 C4FLE9 6419394 IC50 = 150 nM T63966 C4GHT0 6419395 IC50 = 600 nM T63966 C8SAQ1 6419396 IC50 = 600 nM T63966 CP71CL 6419397 IC50 = 350 nM T63966 CSMU27 6425419 IC50 = 87 nM T63966 CUPQ08 6539985 IC50 = 2 nM T63966 CMEZ23 6540005 IC50 = 170 nM T63966 CE47IF 9884465 IC50 = 80 nM T63966 C4R8YV 9884654 IC50 = 132 nM T63966 C76KCF 9950028 IC50 = 470 nM T63966 CG57EC 10047098 IC50 > 50000 nM T63966 CUJR40 10062694 EC50 = 236 nM T63966 C7TA9J 10113568 IC50 = 7.762 nM T63966 CIV15Q 10113978 IC50 = 10 nM T63966 CSGD16 10246246 IC50 > 7000 nM T63966 C1WL8B 10251852 IC50 > 200000 nM T63966 C8RD3V 10301884 IC50 > 33000 nM T63966 C9GK3M 10342546 IC50 = 4 nM T63966 C9ZXG2 10357919 IC50 = 4400 nM T63966 CQB9H7 10389422 IC50 = 11200 nM T63966 C56SVY 10434122 IC50 = 5 nM T63966 C4CV5L 10470475 IC50 = 22000 nM T63966 CIH5K0 11024702 IC50 > 2500 nM T63966 CBOP58 11293798 Ki > 10000 nM T63966 C26BZX 11362471 Ki > 10000 nM T63966 CB45PJ 11362483 IC50 = 73 nM T63966 C25ZCN 11374110 IC50 = 16 nM T63966 CWXB93 11397177 Ki > 10000 nM T63966 CREQ51 11429654 IC50 = 24 nM T63966 CY0A4E 11429729 IC50 = 38 nM T63966 CK3M0T 11495270 IC50 = 5 nM T63966 CL7X4Q 11530963 IC50 = 55 nM T63966 CTG83F 11539329 Ki > 440 nM T63966 CACS26 11561968 Ki > 2000 nM T63966 C0HM3O 11581327 IC50 = 140 nM T63966 C3VUO7 11588815 IC50 = 7 nM T63966 CA2KX0 11590078 IC50 < 3 nM T63966 CMIL86 11590363 Ki > 440 nM T63966 CLWA52 11611374 IC50 = 120 nM T63966 CV71YX 11617549 IC50 = 720 nM T63966 CK34LS 11632737 IC50 = 400 nM T63966 C9T6SC 11640926 Ki > 440 nM T63966 CU0E8O 11690457 Ki > 2000 nM T63966 C45EWD 11723489 IC50 > 7000 nM T63966 CRZ4K6 11724734 IC50 = 66000 nM T63966 CP7AH3 11755812 IC50 = 747 nM T63966 CHR92S 11858109 IC50 = 45 nM T63966 CP2HR6 11948697 IC50 = 4 nM T63966 C60NJV 11948698 IC50 = 10 nM T63966 CC09DE 11955790 IC50 = 47 nM T63966 CDZ1I3 11989153 IC50 = 115.5 nM T63966 CZHQ54 12988783 IC50 = 4 nM T63966 CN14SK 12988792 IC50 = 6 nM T63966 CXRK13 12988793 IC50 = 3 nM T63966 C35LRO 15949471 IC50 = 620 nM T63966 C7LB4I 15949613 IC50 = 15 nM T63966 CFPW41 16007116 Ki > 440 nM T63966 CQI0A5 16043229 IC50 = 14 nM T63966 CZKD04 16043241 IC50 = 79 nM T63966 C9X4TQ 16043242 IC50 = 10 nM T63966 C9TU1O 16046126 IC50 > 1000 nM T63966 C5VPH9 16129448 IC50 = 4220 nM T63966 CW9J7K 16141844 IC50 = 28000 nM T63966 CP3HS4 16220354 IC50 = 2 nM T63966 CDZ31W 16747696 IC50 = 6 nM T63966 CQA78V 18382736 IC50 = 290 nM T63966 C2EBQ5 18382775 IC50 = 18 nM T63966 CZB5L4 18382784 IC50 = 140 nM T63966 C1LUP2 18382794 IC50 = 4 nM T63966 CZ1GR8 18382813 IC50 = 190 nM T63966 C8KJ4R 18382823 IC50 = 250 nM T63966 CZC98J 18382853 IC50 = 130 nM T63966 C5QV1L 18382857 IC50 = 620 nM T63966 C84KLY 18382861 IC50 = 5 nM T63966 CSPD61 18382868 IC50 = 3 nM T63966 CG4BK9 18382875 IC50 = 7 nM T63966 C8BK3Q 18382898 IC50 = 4 nM T63966 CX7F1I 18382902 IC50 = 6 nM T63966 CNE4R0 18382910 IC50 = 56 nM T63966 CML03B 18382946 IC50 = 4 nM T63966 CGXU47 18382956 IC50 = 1410 nM T63966 C5K2DQ 18382971 IC50 = 390 nM T63966 C5BGJ8 18382993 IC50 = 24 nM T63966 CVFU60 18383007 IC50 = 4 nM T63966 CZ90LJ 18383038 IC50 = 770 nM T63966 C5ZF2U 18383051 IC50 = 220 nM T63966 C2R0KU 18383095 IC50 = 500 nM T63966 CBF6H0 18383099 IC50 = 5 nM T63966 C7SQ3Z 18383101 IC50 = 5 nM T63966 CQ7V2F 18383102 IC50 = 3 nM T63966 CL81VC 21100709 IC50 = 3700 nM T63966 CFN6G4 21701597 IC50 = 600 nM T63966 CF6LA9 22478260 IC50 = 650 nM T63966 CMRO51 22478297 IC50 = 750 nM T63966 CBI80A 22664657 IC50 = 22 nM T63966 CP02XA 22664735 IC50 = 14 nM T63966 COB60M 23133320 IC50 = 2000 nM T63966 C9QLP0 23133323 IC50 = 1600 nM T63966 C6JV7W 23400934 IC50 > 7000 nM T63966 CD5S7O 23401001 IC50 > 7000 nM T63966 C0E2GY 23644614 IC50 > 10000 nM T63966 C7E0KL 23644828 IC50 = 4600 nM T63966 C4DBE2 23644829 IC50 > 10000 nM T63966 C72CKL 23644830 IC50 = 310 nM T63966 CC1TK5 23644831 IC50 = 6850 nM T63966 CLP8Y4 23644832 IC50 > 10000 nM T63966 C47NWC 23644833 IC50 > 10000 nM T63966 C2SG8A 23644834 IC50 > 10000 nM T63966 C0JRK8 23644835 IC50 = 5460 nM T63966 CKF20I 23644836 IC50 > 10000 nM T63966 CI64QY 23644837 IC50 = 6410 nM T63966 CL20MD 23644838 IC50 = 840 nM T63966 C4RW2C 23644839 IC50 > 10000 nM T63966 CK2HX6 23644840 IC50 = 160 nM T63966 CM0KD3 23644841 IC50 = 760 nM T63966 CS5HY0 23644842 IC50 > 10000 nM T63966 C4DFA5 23644843 IC50 = 4660 nM T63966 CJ07AS 23644844 IC50 > 10000 nM T63966 CWQX87 23644845 IC50 > 10000 nM T63966 CP3L6Q 23644846 IC50 = 2330 nM T63966 C9ATK1 23644847 IC50 = 5420 nM T63966 C8U6BV 23644848 IC50 = 590 nM T63966 CIZG50 23644849 IC50 = 5320 nM T63966 CKL39U 23644850 IC50 = 720 nM T63966 C4AEC8 23644851 IC50 = 3020 nM T63966 C47LSD 23644852 IC50 = 630 nM T63966 CT4XY0 23644853 IC50 = 750 nM T63966 CG48KV 23644854 IC50 = 3850 nM T63966 C1JM4P 23644855 IC50 > 10000 nM T63966 CU90AF 23644856 IC50 > 10000 nM T63966 C3ZBS6 23644857 IC50 > 10000 nM T63966 CQI9A3 23644858 IC50 = 220 nM T63966 CM7C6T 23644859 IC50 = 760 nM T63966 CCI2M1 23644860 IC50 = 1220 nM T63966 C3Q5FV 23644861 IC50 > 10000 nM T63966 CR83MY 23644862 IC50 > 10000 nM T63966 CCI62P 23644863 IC50 > 10000 nM T63966 CHA4J3 23644864 IC50 > 10000 nM T63966 CB2C4G 23644865 IC50 > 10000 nM T63966 C9O4XE 23644866 IC50 > 10000 nM T63966 C5OQ2T 23644867 IC50 > 10000 nM T63966 C2WAK8 23644868 IC50 > 10000 nM T63966 C21APY 23644869 IC50 > 10000 nM T63966 CA92DC 23644870 IC50 = 440 nM T63966 CZ9L7X 23644871 IC50 > 10000 nM T63966 CK42DF 23644872 IC50 = 770 nM T63966 CO06PR 23644873 IC50 = 220 nM T63966 CH4S6V 23644874 IC50 = 270 nM T63966 CY9FT0 23644875 IC50 = 480 nM T63966 CEB43Q 23644876 IC50 > 10000 nM T63966 C2RN3L 23644877 IC50 = 730 nM T63966 C5XWJ8 23644878 IC50 = 560 nM T63966 CAZL79 23644879 IC50 = 320 nM T63966 CJR51Z 23644880 IC50 = 810 nM T63966 CGBW01 23644881 IC50 = 930 nM T63966 CUIT84 23644882 IC50 = 840 nM T63966 CZH4Q1 23644883 IC50 = 530 nM T63966 C3Y5BN 23644884 IC50 = 470 nM T63966 CSOG87 23644885 IC50 = 670 nM T63966 CT81BV 23644886 IC50 = 260 nM T63966 CM9YD6 23644887 IC50 = 710 nM T63966 CW20PU 23644888 IC50 = 740 nM T63966 C2ODX8 23644889 IC50 = 1070 nM T63966 C9C5LQ 23644890 IC50 = 500 nM T63966 C7BGR4 23644891 IC50 > 10000 nM T63966 C6P1JN 23644892 IC50 > 10000 nM T63966 CIJ3K8 23644893 IC50 = 270 nM T63966 CV2MF6 23644894 IC50 = 180 nM T63966 CET2G3 23644895 IC50 = 120 nM T63966 CPX58K 23644896 IC50 = 140 nM T63966 C3U9RZ 23644897 IC50 > 10000 nM T63966 CSFK63 23646936 IC50 = 138.04 nM T63966 CEN96M 23646937 IC50 = 1737.8 nM T63966 CJ5H1Z 23646938 IC50 = 7.079 nM T63966 CIP7T2 23646939 IC50 = 186.21 nM T63966 CL4ST0 23646940 IC50 = 331.13 nM T63966 C4E2OX 23646941 IC50 = 446.68 nM T63966 CI32JB 23646942 IC50 = 23.99 nM T63966 C2S5ZM 23661662 Ki = 110 nM T63966 CYWG82 23729145 IC50 > 1000 nM T63966 CHU49V 24757938 IC50 = 0.5 nM T63966 CY8X0J 24811794 Ki > 10000 nM T63966 C43HWQ 24883287 IC50 > 10000 nM T63966 C8DA5Q 24883334 IC50 = 10000 nM T63966 CY8L7E 24896769 IC50 > 10000 nM T63966 CUIG07 24905422 IC50 = 300 nM T63966 COB43M 25014810 IC50 = 34000 nM T63966 CRO0Y8 25022735 IC50 > 200000 nM T63966 C72AJM 25022736 IC50 > 200000 nM T63966 C0B7RT 25057409 IC50 > 10000 nM T63966 C2ICS7 25065806 IC50 = 591 nM T63966 CTV54O 25123227 IC50 = 3.6 nM T63966 C1IYN7 25127854 IC50 = 6.4 nM T63966 CKD14B 25127856 IC50 = 33 nM T63966 CJBX60 25128180 IC50 = 56 nM T63966 CC5SD9 25128181 IC50 = 69 nM T63966 COB9G8 25181586 IC50 = 118100 nM T63966 C8IJB9 25218207 IC50 = 160100 nM T63966 CC71QJ 27666048 IC50 > 100000 nM T63966 C8B6TY 42628503 EC50 < 500 nM T63966 CHQ24O 44156904 IC50 = 72 nM T63966 CI50DJ 44156905 IC50 = 130 nM T63966 CNH12Z 44156906 IC50 = 110 nM T63966 C1V7TM 44156907 IC50 = 170 nM T63966 CT19KO 44156908 IC50 = 210 nM T63966 C2W0XB 44156915 IC50 = 66 nM T63966 CIM89D 44157074 IC50 = 130 nM T63966 CEL61X 44229839 IC50 > 10000 nM T63966 CKD14Y 44316725 IC50 = 3 nM T63966 CM2A1F 44316744 IC50 = 4 nM T63966 CLJ2P3 44316765 IC50 = 43 nM T63966 CK9L3S 44316797 IC50 = 2 nM T63966 C8IAY4 44316957 IC50 = 22 nM T63966 CD69PV 44317138 IC50 = 17 nM T63966 C7AR0V 44317156 IC50 = 2000 nM T63966 C9RY8G 44317213 IC50 > 2500 nM T63966 CQN1R8 44331899 IC50 = 23000 nM T63966 CYV2D7 44368815 IC50 = 130 nM T63966 C4Q6AU 44408662 IC50 = 560 nM T63966 CQS1C8 44408663 IC50 = 1260 nM T63966 CO9Y5V 44408666 IC50 = 670 nM T63966 CMK9U8 44408667 IC50 > 10000 nM T63966 CE69KV 44408690 IC50 > 10000 nM T63966 CZ7EC3 44408694 IC50 = 490 nM T63966 CG8FQ3 44408695 IC50 = 590 nM T63966 COKT15 44408845 IC50 > 10000 nM T63966 C0UZB8 44408850 IC50 > 10000 nM T63966 CJC51Y 44408863 IC50 = 890 nM T63966 CKT3D9 44408868 IC50 = 770 nM T63966 CZU6Y2 44408869 IC50 = 460 nM T63966 C6E9XY 44408879 IC50 = 510 nM T63966 CH2V8K 44408916 IC50 = 160 nM T63966 CHZ7R4 44408923 IC50 = 590 nM T63966 C6DKJ9 44408924 IC50 = 440 nM T63966 CB71IO 44408930 IC50 = 1470 nM T63966 C04IOD 44408931 IC50 > 10000 nM T63966 CIQ75Y 44408972 IC50 > 10000 nM T63966 CR4X5E 44408975 IC50 > 10000 nM T63966 C5VN0R 44409048 IC50 > 10000 nM T63966 CJE32H 44409051 IC50 = 340 nM T63966 CSZ9Y5 44409052 IC50 = 300 nM T63966 CZJP10 44409058 IC50 = 220 nM T63966 CC9NV5 44409070 IC50 > 10000 nM T63966 CNT4R5 44409071 IC50 > 10000 nM T63966 CT4O5I 44409087 IC50 = 740 nM T63966 CJIC91 44409090 IC50 = 570 nM T63966 C0C5FS 44409091 IC50 > 10000 nM T63966 CD3Q8H 44409100 IC50 > 10000 nM T63966 C4WDI5 44409106 IC50 = 220 nM T63966 CI71ZK 44409142 IC50 > 10000 nM T63966 CBX37N 44409151 IC50 = 950 nM T63966 C2M8WP 44409154 IC50 = 770 nM T63966 C4JH7R 44409166 IC50 = 1140 nM T63966 CRW9G6 44409167 IC50 = 2530 nM T63966 C3Z9HC 44409172 IC50 > 10000 nM T63966 CC5U3T 44409175 IC50 = 3310 nM T63966 CF75LM 44409176 IC50 > 10000 nM T63966 C5S6UA 44409188 IC50 > 10000 nM T63966 C26DKP 44409192 IC50 = 760 nM T63966 CRN61C 44409200 IC50 = 340 nM T63966 C1E9AZ 44409202 IC50 > 10000 nM T63966 CY80ID 44409203 IC50 > 10000 nM T63966 C2ZAL9 44409207 IC50 = 1470 nM T63966 CKM2X3 44409224 IC50 = 1160 nM T63966 CX0DN5 44409262 IC50 = 610 nM T63966 C05SDW 44409266 IC50 = 540 nM T63966 C21FOV 44409267 IC50 = 440 nM T63966 CUK1I5 44409271 IC50 = 1250 nM T63966 C16QCJ 44409285 IC50 = 260 nM T63966 C1W7AS 44409294 IC50 = 410 nM T63966 CC79ES 44409305 IC50 > 10000 nM T63966 CH15MA 44409306 IC50 > 10000 nM T63966 C29AMO 44409313 IC50 > 10000 nM T63966 CGO3A8 44409320 IC50 = 690 nM T63966 CBM5T2 44409324 IC50 = 340 nM T63966 C8WJ1O 44409325 IC50 = 490 nM T63966 C5SH2J 44409329 IC50 = 180 nM T63966 CMGA85 44409431 IC50 = 360 nM T63966 CS8YQ2 44414316 IC50 = 36 nM T63966 C7KZV2 44414322 IC50 = 601 nM T63966 CJM06T 44414347 IC50 = 970 nM T63966 CBZ2X3 44414348 IC50 = 592 nM T63966 C84DVH 44414371 IC50 = 3842 nM T63966 C32UEI 44414376 IC50 = 2897 nM T63966 C45PBG 44414394 IC50 = 131 nM T63966 CD1I5Y 44414395 IC50 = 2263 nM T63966 CF2JA5 44414419 IC50 = 59 nM T63966 C3G2FJ 44414460 IC50 = 3785 nM T63966 C6YL5H 44414486 IC50 = 2056 nM T63966 C5RTK0 44414527 IC50 = 38 nM T63966 CRL1C4 44414547 IC50 = 1590 nM T63966 C0MZ7P 44414549 IC50 = 64 nM T63966 C3SYD7 44414595 IC50 = 2824 nM T63966 CP6TZ2 44414596 IC50 = 3615 nM T63966 C6I8TW 44414597 IC50 = 25 nM T63966 CIQA35 44414621 IC50 = 38 nM T63966 CUW8C1 44414632 IC50 = 1351 nM T63966 C06UCM 44414633 IC50 = 20 nM T63966 CQB17H 44414646 IC50 = 33 nM T63966 CLD07U 44414647 IC50 = 19 nM T63966 CTAZ73 44414648 IC50 = 83 nM T63966 C1XCW7 44414659 IC50 > 50000 nM T63966 C1TR2Y 44414666 IC50 = 1668 nM T63966 CBY7D9 44414679 IC50 = 39 nM T63966 CO14UX 44414683 IC50 = 24996 nM T63966 C1LZ9S 44414695 IC50 = 11483 nM T63966 C0JF1Z 44414779 IC50 = 75 nM T63966 C0THE4 44414816 IC50 = 2275 nM T63966 CRF01G 44414847 IC50 > 50000 nM T63966 CXV94N 44414848 IC50 = 14581 nM T63966 CUI2N3 44414867 IC50 = 863 nM T63966 C8LH5Q 44414868 IC50 = 27894 nM T63966 CD13BL 44414880 IC50 = 4201 nM T63966 CTCM71 44414881 IC50 = 4953 nM T63966 C5WGQ0 44421704 IC50 = 4718 nM T63966 CF34KY 44421705 IC50 = 44 nM T63966 CETQ79 44427518 IC50 > 50000 nM T63966 COPG94 44427519 IC50 > 10000 nM T63966 CND24H 44431888 IC50 > 10000 nM T63966 CJHD30 44431889 IC50 > 10000 nM T63966 C5X8IO 44431890 IC50 = 97 nM T63966 CF31BX 44431891 IC50 > 10000 nM T63966 C6DME5 44431892 IC50 > 10000 nM T63966 CK1AS2 44431893 IC50 > 10000 nM T63966 CJ73EF 44431894 IC50 > 10000 nM T63966 C3SG5E 44431895 IC50 > 10000 nM T63966 C6VZ8W 44431896 IC50 > 10000 nM T63966 C6YL7I 44431897 IC50 = 380 nM T63966 CU4MN1 44431898 IC50 = 220 nM T63966 CTR14P 44431899 IC50 = 190 nM T63966 C8OWB5 44431900 IC50 = 450 nM T63966 C2IJ4Q 44431901 IC50 = 320 nM T63966 C2Y4XS 44431902 IC50 = 590 nM T63966 CME54X 44431903 IC50 = 440 nM T63966 C0KM8Y 44431904 IC50 = 2250 nM T63966 C5B2EM 44431905 IC50 = 5250 nM T63966 C79PXH 44431906 IC50 > 10000 nM T63966 CRC6N1 44431907 IC50 = 380 nM T63966 C46YKU 44431908 IC50 > 10000 nM T63966 CJSK07 44431909 IC50 > 10000 nM T63966 C36QDE 44431910 IC50 = 2330 nM T63966 CET6B3 44431911 IC50 = 980 nM T63966 CUM12J 44431912 IC50 = 860 nM T63966 CB73ES 44431913 IC50 = 1230 nM T63966 C35AGI 44431914 IC50 = 1220 nM T63966 C75NGZ 44431915 IC50 = 2250 nM T63966 C6ANT8 44431916 IC50 > 10000 nM T63966 CD4QB5 44431917 IC50 > 10000 nM T63966 CPRX24 44431918 IC50 > 10000 nM T63966 CL85AI 44431919 IC50 > 10000 nM T63966 CP68DH 44431920 IC50 = 940 nM T63966 CDX70N 44431921 IC50 = 790 nM T63966 CXQ4K6 44431922 IC50 = 4270 nM T63966 C8Q1XM 44431925 IC50 = 3860 nM T63966 C9NY4F 44431927 IC50 = 4560 nM T63966 C6C5GM 44431928 IC50 > 10000 nM T63966 CTL31N 44431930 IC50 > 10000 nM T63966 C58POW 44431932 IC50 > 10000 nM T63966 CZT4Y3 44431935 IC50 = 890 nM T63966 C1O5QH 44431936 IC50 = 1080 nM T63966 CGR4F6 44431939 IC50 = 3880 nM T63966 C6EL0U 44431940 IC50 > 10000 nM T63966 C1Z6NQ 44431941 IC50 > 10000 nM T63966 CF72BI 44432051 IC50 > 10000 nM T63966 CA98KR 44432441 IC50 > 10000 nM T63966 C0YU5D 44439355 IC50 > 10000 nM T63966 C4UO8C 44439356 IC50 = 2270 nM T63966 C0IXS5 44439357 IC50 = 1680 nM T63966 CL7Q0Z 44439358 IC50 > 10000 nM T63966 CGSR93 44439359 IC50 = 650 nM T63966 CT3B4P 44439360 IC50 = 1980 nM T63966 CWS7D3 44439361 IC50 = 1150 nM T63966 COYR48 44439362 IC50 = 760 nM T63966 C1PIW8 44439363 IC50 = 250 nM T63966 CZP54X 44439364 IC50 = 2060 nM T63966 C1CB7D 44439365 IC50 = 180 nM T63966 C3QH1P 44439366 IC50 = 3770 nM T63966 C9GH4W 44439367 IC50 = 4290 nM T63966 CLME26 44439368 IC50 = 5570 nM T63966 C1S3IP 44439369 IC50 = 230 nM T63966 C5YT3N 44439448 IC50 = 5730 nM T63966 CK1O5J 44439449 IC50 = 950 nM T63966 C9XE4V 44439450 IC50 = 290 nM T63966 C75DRT 44439451 IC50 = 370 nM T63966 CXI3B5 44439452 IC50 = 210 nM T63966 CZ5T6X 44439453 IC50 = 580 nM T63966 C4C0XH 44439454 IC50 = 740 nM T63966 C37IHP 44439455 IC50 = 340 nM T63966 C13TLQ 44439457 IC50 = 210 nM T63966 CZM4Y0 44439458 IC50 = 840 nM T63966 CO29LB 44439459 IC50 = 650 nM T63966 CY76DC 44439460 IC50 > 10000 nM T63966 C35RTN 44439461 IC50 = 5290 nM T63966 CU2SG9 44439462 IC50 > 10000 nM T63966 CG0A7Z 44439463 IC50 > 10000 nM T63966 C4R8HQ 44439464 IC50 = 750 nM T63966 CDQ6K8 44439465 IC50 = 280 nM T63966 C6DQV9 44439466 IC50 = 730 nM T63966 CVP1S9 44439467 IC50 = 2060 nM T63966 C5VL4O 44439468 IC50 = 4580 nM T63966 CS49IA 44439469 IC50 = 2060 nM T63966 CN65DW 44439470 IC50 = 130 nM T63966 C4BJI2 44439471 IC50 = 290 nM T63966 CTU07B 44439472 IC50 > 10000 nM T63966 C1WFV5 44439475 IC50 > 10000 nM T63966 CE1U3I 44439478 IC50 = 5570 nM T63966 CBC3V5 44439479 IC50 = 280 nM T63966 CQ9Y7K 44439480 IC50 = 1130 nM T63966 C97RIN 44439481 IC50 = 210 nM T63966 CI75KD 44439482 IC50 = 250 nM T63966 C03YPU 44439484 IC50 = 350 nM T63966 CL7KY8 44439487 IC50 = 840 nM T63966 CYU6S0 44439495 IC50 = 1120 nM T63966 C05LUV 44439496 IC50 = 660 nM T63966 C9J0IC 44439497 IC50 = 330 nM T63966 C6A3OB 44439499 IC50 = 1560 nM T63966 CH6FM2 44439501 IC50 = 370 nM T63966 C09HPL 44439502 IC50 = 2120 nM T63966 C98OAT 44439503 IC50 = 5660 nM T63966 CA81EQ 44439504 IC50 > 10000 nM T63966 CLFS52 44439505 IC50 > 10000 nM T63966 C8YZ0F 44439506 IC50 = 280 nM T63966 C9M4SR 44439507 IC50 = 440 nM T63966 C09PNG 44439508 IC50 > 10000 nM T63966 C7F1SN 44439509 IC50 > 10000 nM T63966 C25SEZ 44439510 IC50 = 5800 nM T63966 CR5K0Q 44439511 IC50 = 940 nM T63966 CQ0E2J 44439512 IC50 = 3270 nM T63966 COC5E7 44439513 IC50 = 560 nM T63966 CQO50A 44439514 IC50 = 970 nM T63966 C9KC5D 44439515 IC50 = 1190 nM T63966 CJL03B 44439516 IC50 = 4230 nM T63966 CU4O8W 44439517 IC50 = 870 nM T63966 C14MTJ 44440231 IC50 = 3470 nM T63966 CA86YP 44440232 IC50 = 3080 nM T63966 COK21X 44440233 IC50 = 17570 nM T63966 CYMN10 44440242 IC50 = 370 nM T63966 C96ARW 44440243 IC50 = 240 nM T63966 CGL0R4 44440244 IC50 = 270 nM T63966 CQI8S3 44440245 IC50 = 290 nM T63966 CZM08I 44440246 IC50 = 30 nM T63966 C4O8NF 44440247 IC50 = 450 nM T63966 C1DAU0 44440248 IC50 = 290 nM T63966 C93TBM 44440249 IC50 = 80 nM T63966 C6VLC0 44440250 IC50 = 90 nM T63966 CO37FE 44440251 IC50 = 70 nM T63966 C6T0IK 44440252 IC50 = 50 nM T63966 CJ05OC 44440253 IC50 = 710 nM T63966 CGV37F 44440254 IC50 = 710 nM T63966 C5JUV3 44440256 IC50 = 136 nM T63966 CFB56S 44440259 IC50 = 20 nM T63966 CEW9G2 44440261 IC50 = 153 nM T63966 C5R4QE 44442729 Ki = 1600 nM T63966 CGC76I 44442730 Ki > 10000 nM T63966 CJM6N5 44442731 Ki > 10000 nM T63966 CH2FS6 44442732 Ki > 10000 nM T63966 CZ7FC6 44442733 Ki > 10000 nM T63966 C6PNZ4 44442734 Ki = 910 nM T63966 C8N1EQ 44442735 Ki = 1710 nM T63966 C26EVP 44442736 Ki = 1900 nM T63966 C0S6PN 44442737 Ki = 2900 nM T63966 CAZ5O7 44442738 Ki = 350 nM T63966 CM9XW1 44442739 Ki = 1500 nM T63966 CFOH51 44442740 Ki > 10000 nM T63966 CX10DZ 44442742 Ki = 1400 nM T63966 CN12IA 44442744 Ki > 10000 nM T63966 C0DOP6 44442745 Ki = 920 nM T63966 C3PGF0 44444786 IC50 = 121000 nM T63966 CMJ6Y5 44444788 IC50 = 31100 nM T63966 C6JZ5E 44444796 IC50 = 93000 nM T63966 CK9D5S 44444803 IC50 = 162000 nM T63966 C4YMI9 44447890 IC50 = 8 nM T63966 C6I1TW 44560803 IC50 = 3 nM T63966 CTI4C0 44564574 IC50 = 510 nM T63966 CE3MP5 44564575 IC50 = 1130 nM T63966 CFM8P1 44564576 IC50 = 650 nM T63966 CPIR15 44564600 IC50 = 860 nM T63966 CP63RZ 44564651 IC50 > 10000 nM T63966 C5P0EK 44564652 IC50 > 10000 nM T63966 CTF0V2 44564653 IC50 > 10000 nM T63966 CIVF90 44564688 IC50 > 10000 nM T63966 C21HAM 44564690 IC50 > 10000 nM T63966 C1JH3T 44564727 IC50 > 10000 nM T63966 CTK29Y 44565090 IC50 > 10000 nM T63966 CER4M3 44565091 IC50 > 10000 nM T63966 CB3U0T 44565092 IC50 > 10000 nM T63966 C6F0SN 44565141 IC50 > 10000 nM T63966 CXS46L 44565142 IC50 = 130 nM T63966 CI5D3M 44565143 IC50 = 660 nM T63966 CKE2W7 44565144 IC50 = 1130 nM T63966 CP6F5U 44565194 IC50 = 250 nM T63966 C1XHB9 44565195 IC50 = 530 nM T63966 C7P9CB 44565196 IC50 = 640 nM T63966 CVT9H8 44565197 IC50 = 650 nM T63966 CYUI08 44566353 IC50 = 65000 nM T63966 C0N4ZA 44577698 IC50 = 1900 nM T63966 C4BFY1 44577740 IC50 = 460 nM T63966 C4Q3YF 44577741 IC50 = 270 nM T63966 C5WOE2 44586449 IC50 = 45100 nM T63966 C0VF8M 44586450 IC50 = 31800 nM T63966 C4K7NP 44586451 IC50 = 32700 nM T63966 C1JNR5 44586452 IC50 = 7800 nM T63966 C6T8UP 44586490 IC50 > 200000 nM T63966 CU95NI 44586526 IC50 > 200000 nM T63966 CBK9R3 44586527 IC50 > 200000 nM T63966 CA18IW 44586528 IC50 > 200000 nM T63966 C0YSZ2 44586577 IC50 > 200000 nM T63966 CGQR60 44586767 IC50 = 84000 nM T63966 CVRQ96 44586768 IC50 > 100000 nM T63966 C05HTO 44586769 IC50 = 100000 nM T63966 CX0R8V 44586770 IC50 = 96000 nM T63966 CQA2K1 44586794 IC50 > 100000 nM T63966 CH67VY 44586829 IC50 > 100000 nM T63966 C0HOF8 44586830 IC50 = 5200 nM T63966 C86ADQ 44586832 IC50 > 100000 nM T63966 CZAF65 44586833 IC50 > 100000 nM T63966 CWP37F 44586834 IC50 = 79000 nM T63966 CT5HM0 44586867 IC50 = 23000 nM T63966 CGK6C7 44586868 IC50 > 100000 nM T63966 C70DAO 44586869 IC50 = 68000 nM T63966 C2JIZ9 44586870 IC50 > 100000 nM T63966 CYU2G3 44586896 IC50 > 100000 nM T63966 C7G6KH 44586897 IC50 = 31000 nM T63966 C4L9BF 44586898 IC50 > 100000 nM T63966 CM45ZR 44586899 IC50 > 100000 nM T63966 CVU93G 44586900 IC50 > 100000 nM T63966 CMV3W2 44586901 IC50 > 100000 nM T63966 CV2W4P 44586928 IC50 > 100000 nM T63966 C95XRW 44586929 IC50 > 100000 nM T63966 CCT91D 44586930 IC50 = 36000 nM T63966 CJ4HT0 44587324 IC50 > 100000 nM T63966 CD56YX 44587325 IC50 > 100000 nM T63966 C4KW0O 44587326 IC50 = 77000 nM T63966 CX3O7R 44590991 IC50 = 2510 nM T63966 CBJ92M 44590992 IC50 = 700 nM T63966 CDG2S0 44590993 IC50 > 10000 nM T63966 CF78DX 44590994 IC50 > 10000 nM T63966 CKBN26 44590995 IC50 > 10000 nM T63966 CE91VG 44591030 IC50 = 330 nM T63966 CAI2X9 44591117 IC50 = 580 nM T63966 CD51XN 44591118 IC50 > 10000 nM T63966 CH0O2G 44591119 IC50 > 10000 nM T63966 C90IVK 44591355 IC50 > 10000 nM T63966 CE4G8R 44591356 IC50 > 10000 nM T63966 CN39VL 44591357 IC50 = 250 nM T63966 C5JYA9 44591358 IC50 > 10000 nM T63966 C7EOZ3 44591359 IC50 > 10000 nM T63966 C9WXA4 44591374 IC50 = 260 nM T63966 C9C8AH 44591375 IC50 = 1230 nM T63966 C4E3NV 44591376 IC50 = 310 nM T63966 CUZG74 44591377 IC50 = 610 nM T63966 C1JOA9 44591378 IC50 = 250 nM T63966 C9YV4O 44591404 IC50 = 55 nM T63966 C0AWD1 44591405 IC50 = 260 nM T63966 C6EBW0 44591406 IC50 > 10000 nM T63966 C5XJ2N 44591407 IC50 = 380 nM T63966 CZ8F6B 44591439 IC50 = 980 nM T63966 CL7RC8 44591440 IC50 = 1800 nM T63966 C0T1RY 44591441 IC50 = 750 nM T63966 CL1TJ4 44591442 IC50 = 190 nM T63966 CQ9VS5 44591443 IC50 = 670 nM T63966 CY3HW5 46224684 IC50 = 9000 nM T63966 C2P9QO 46228508 IC50 = 1530 nM T63966 C6E5PY 46228822 IC50 = 4160 nM T63966 C3T8AM 46228951 IC50 = 4840 nM T63966 CYZV41 46231219 IC50 = 150 nM T63966 C7J5UP 46231220 IC50 = 69.4 nM T63966 CC96GZ 46231221 IC50 = 72.4 nM T63966 CQN86H 46831064 IC50 = 101000 nM T63966 CFR1C6 46845026 IC50 > 300000 nM T63966 C5WC9K 46871765 IC50 = 2100 nM T63966 CLS29B 46872626 IC50 > 10000 nM T63966 CA57MX 46886970 IC50 = 70900 nM T63966 CRGH62 46886971 IC50 = 162900 nM T63966 C68AGR 46886972 IC50 = 156100 nM T63966 CP32GW 46886973 IC50 > 300000 nM T63966 C48JWD 46886974 IC50 > 300000 nM T63966 C7H3MD 46887038 IC50 = 157000 nM T63966 C40NOR 46887039 IC50 = 163100 nM T63966 C7I4SB 46887074 IC50 > 300000 nM T63966 CI5QX2 46887110 IC50 > 300000 nM T63966 C0Q7NG 46887111 IC50 = 150900 nM T63966 CU15AN 46887112 IC50 > 300000 nM T63966 CD90BV 46887113 IC50 > 300000 nM T63966 CH3O9K 46887255 IC50 = 129400 nM T63966 C7NUT3 46887298 IC50 = 142300 nM T63966 CWV65D 46887299 IC50 > 200000 nM T63966 CH5BZ6 46887300 IC50 > 200000 nM T63966 C20UCB 46887348 IC50 = 164300 nM T63966 C0KEG5 46887349 IC50 > 200000 nM T63966 CY59RB 46887397 IC50 = 223800 nM T63966 CW7AR1 46889887 IC50 = 28 nM T63966 CMNK35 46889911 IC50 = 16 nM T63966 C0WYM1 46898022 IC50 = 10000 nM T63966 CHSF07 49806372 IC50 > 1000 nM T63966 CY90BD 49818230 IC50 = 1275 nM T63966 CB0S2P 49842666 IC50 = 51000 nM T63966 CAI20B 49842778 IC50 = 33000 nM T63966 CRA74I 49842779 IC50 > 100000 nM T63966 CB5O0I 49860186 IC50 = 25 nM T63966 C9W6SO 49860190 IC50 = 550 nM T63966 CQ3KU9 50899556 IC50 = 470 nM T63966 CS9G6E 50997096 IC50 > 10000 nM T63966 C3LB5V 52941849 IC50 = 74 nM T63966 CW2X5E 52944268 IC50 = 2 nM T63966 C9PX2J 52945752 IC50 = 4 nM T63966 CL4ED3 52945753 IC50 = 40 nM T63966 CIR3Q0 52947964 IC50 > 10000 nM T63966 C09SDH 53257410 IC50 = 3200 nM T63966 C2P3OT 53316977 IC50 > 100000 nM T63966 CB2KU7 53318682 IC50 = 102700 nM T63966 C5SU2K 53320001 IC50 = 91600 nM T63966 CFX89P 53321301 IC50 = 36500 nM T63966 CK9R3I 53322631 IC50 = 61200 nM T63966 CDV5Y7 53323499 IC50 = 76800 nM T63966 CZY0J7 53323592 IC50 = 15000 nM T63966 CRT5F8 53325256 IC50 = 109500 nM T63966 CNPM14 53341082 IC50 > 3000 nM T63966 CE8OA7 53357593 IC50 = 310 nM T63966 CBK9Q6 53357848 IC50 > 10000 nM T63966 C8NA4L 53384644 IC50 > 30000 nM T63966 C8AB1J 54759606 Ki = 1100 nM T63966 C1ST0I 56656325 IC50 = 93200 nM T63966 C8IZ4J 56659759 IC50 > 1000000 nM T63966 CPG0I4 56659823 IC50 > 1000 nM T63966 C4UPH5 56659824 IC50 = 270 nM T63966 CVDT38 56659825 IC50 > 1000000 nM T63966 C3A7HL 56663233 IC50 > 1000000 nM T63966 CY12ML 56663288 IC50 = 570 nM T63966 CK53GA 56663289 IC50 > 1000 nM T63966 CY2RD1 56663290 IC50 > 1000 nM T63966 C6XVT5 56666663 IC50 > 1000000 nM T63966 C1HTO5 56670140 IC50 = 2610 nM T63966 CC3J1A 56673651 IC50 = 210 nM T63966 C4TD2Q 56673654 IC50 = 40 nM T63966 CGN54D 56676922 IC50 > 1000000 nM T63966 CU0M8W 56676973 IC50 = 140 nM T63966 CH5R3Q 56676974 IC50 > 1000 nM T63966 CUD53B 56676975 IC50 > 1000 nM T63966 CO2GI9 56676977 IC50 > 1000000 nM T63966 CFS43O 56680303 IC50 > 1000 nM T63966 C5RK1U 56680304 IC50 > 1000 nM T63966 CSX3Y4 56683569 IC50 > 1000000 nM T63966 CVM7U4 56683624 IC50 = 420 nM T63966 CBW28D 56683625 IC50 > 1000 nM T63966 CR50TJ 56835147 IC50 = 1920 nM T63966 C2ML5S 56837168 IC50 = 205 nM T63966 CCW89V 56932477 IC50 = 364.5 nM T63966 C7U9SL 56951304 IC50 = 19200 nM T63966 C0GQ9I 56951305 IC50 > 200000 nM T63966 C5YT6A 56951306 IC50 = 31100 nM T63966 CB03EH 56951307 IC50 > 200000 nM T63966 CP58NG 56954518 IC50 = 46 nM T63966 C4YFJ5 57384105 IC50 = 126300 nM T63966 CV9RW5 57384106 IC50 = 156500 nM T63966 CR4T2Y 57391283 IC50 > 200000 nM T63966 CBL74E 57392425 IC50 = 15200 nM T63966 CG18LI 57394786 IC50 = 138100 nM T63966 CEDP89 57394787 IC50 = 150000 nM T63966 CP6W4C 57394879 IC50 = 99300 nM T63966 CVR13L 57394880 IC50 = 79900 nM T63966 CA4Q3Y 57395925 IC50 = 185600 nM T63966 CUGP85 57396545 IC50 = 50800 nM T63966 CBUP96 57396646 IC50 = 129300 nM T63966 CXJ68F 57398331 IC50 = 118600 nM T63966 C14ANY 57398417 IC50 > 200000 nM T63966 CZSM95 57412684 IC50 > 1000 nM T63966 CE59QS 57505507 IC50 = 7.4 nM T63966 C8P6RD 57505528 IC50 = 8.4 nM T63966 C8R4FE 57991377 IC50 = 910.5 nM T63966 C6BPR2 58985201 IC50 > 50000 nM T63966 C1MR8Q 60097495 IC50 > 1000 nM T63966 C7MLW5 60182318 IC50 = 0.1 nM T63966 CN3W2C 60199004 IC50 > 1000 nM T63966 C9ZCT2 62705065 IC50 > 1000 nM T63966 C10AMI 66553589 IC50 = 8160 nM T63966 C37NKO 67129970 IC50 > 10000 nM T63966 CK80LJ 67130050 IC50 > 10000 nM T63966 CQ97ZW 67161103 IC50 = 166 nM T63966 CNP52W 67163022 IC50 = 25 nM T63966 CV63UL 67240318 IC50 > 10000 nM T63966 C7GRV2 68755406 IC50 > 10000 nM T63966 CECZ23 70654418 IC50 > 1000 nM T63966 C4BS5T 70654492 IC50 = 70 nM T63966 CKP9E6 70654499 IC50 = 320 nM T63966 CEXK08 70654539 IC50 > 1000 nM T63966 C0AP6Q 70654571 IC50 > 1000 nM T63966 CRVS29 70654613 IC50 > 1000 nM T63966 COV46X 70654614 IC50 = 350 nM T63966 CP0O5A 70654694 IC50 > 1000 nM T63966 C9QS6O 70654709 IC50 = 54 nM T63966 CC0S3D 70654753 IC50 > 1000 nM T63966 CWE94C 70654840 IC50 = 590 nM T63966 CS6I4T 70654868 IC50 = 200 nM T63966 CGU2P6 70654923 IC50 > 1000 nM T63966 C59APG 70654958 IC50 = 420 nM T63966 C6EK1V 70654997 IC50 = 290 nM T63966 CJAI19 70655010 IC50 = 250 nM T63966 CX3V5C 70655056 IC50 = 320 nM T63966 CW8XC7 70655063 IC50 > 1000 nM T63966 CUYK36 70655070 IC50 = 370 nM T63966 CNQ56Y 70657170 IC50 = 180 nM T63966 C5U0EL 70661438 IC50 > 1000 nM T63966 C03CKB 70661448 IC50 = 20 nM T63966 CGA43T 70690710 IC50 = 82 nM T63966 C6U8HO 70693451 IC50 = 613 nM T63966 CEBO91 71452977 IC50 > 10000 nM T63966 CKT60L 71455860 Ki = 14 nM T63966 CVP2J9 71521862 IC50 = 15000 nM T63966 C5OBF0 71525245 IC50 = 93600 nM T63966 CJX73B 71525246 IC50 > 200000 nM T63966 CCN90I 71525247 IC50 = 103100 nM T63966 CY6JA9 71525248 IC50 > 200000 nM T63966 CGQJ60 71525249 IC50 > 200000 nM T63966 CMKD15 71525283 IC50 > 200000 nM T63966 C3OJ6R 71525284 IC50 > 200000 nM T63966 CP5Q2U 71525285 IC50 = 156300 nM T63966 CZ8N0J 71525286 IC50 = 129600 nM T63966 CG31MI 71525287 IC50 = 189600 nM T63966 C1BCX0 71579696 IC50 > 1000 nM T63966 CZ31PU 71583657 IC50 > 10000 nM T63966 CB64IQ 72194525 IC50 = 19.8 nM T63966 CQXZ13 72700883 Ki = 2400 nM T63966 C60TUV 72737208 IC50 > 10000 nM T63966 CJ3WA6 72737404 IC50 > 10000 nM T63966 CVIU05 73345638 IC50 = 96000 nM T63966 CV21FR 73349643 IC50 = 1000 nM T63966 CAUF10 73351741 IC50 = 151000 nM T63966 C9TMA1 73352657 IC50 = 200 nM T63966 CYJ2B0 73356269 IC50 = 19400 nM T63966 C1TB7K 73356270 IC50 = 22900 nM T63966 CYQ8K1 73357210 IC50 = 20 nM T63966 CVNW01 73386831 IC50 > 1000 nM T63966 CGDB30 74538658 IC50 = 20 nM T63966 CH8W7D 77461036 IC50 > 1000 nM T63966 CCJ43A 86302281 IC50 > 10000 nM T63966 CB5NJ4 86302541 IC50 = 35.1 nM T63966 CPG3A5 86302574 IC50 > 30000 nM T63966 CX29IY 90655145 IC50 > 10000 nM T63966 CRL86F 90665697 IC50 > 1000 nM T63966 C9V6FU 90666397 IC50 > 1000 nM T63966 C5Q8VO 90666398 IC50 > 1000 nM T63966 CIB1E8 90666399 IC50 > 1000 nM T63966 C08ANK 90666400 IC50 > 1000 nM T63966 CL0KH2 90666401 IC50 > 1000 nM T63966 C9XI3E 90666402 IC50 > 1000 nM T63966 CLF29C 90666403 IC50 > 1000 nM T63966 CU9XB7 90666404 IC50 > 1000 nM T63966 CCL19D 90666405 IC50 > 1000 nM T63966 CYVM38 90666406 IC50 > 1000 nM T63966 CMY4T0 90666407 IC50 > 1000 nM T63966 CNE54X 90666408 IC50 > 1000 nM T63966 C8U0ZH 118737468 IC50 = 11.2 nM T63966 C08KEM 122179540 IC50 = 3000 nM T63966 CG0RP7 122179547 IC50 = 2600 nM T63966 C1A0SQ 122179548 IC50 = 5300 nM T63966 C4X7SD 122192466 IC50 = 2826 nM T63966 CNX0Q2 122193763 IC50 = 5750 nM T63966 CWV0C3 122193764 IC50 > 10000 nM T63966 CSG98Y 122193765 IC50 = 7150 nM T63966 CCLQ75 122193769 IC50 = 650 nM T63966 CXDR48 122193770 IC50 = 1080 nM T63966 CPA8C5 122193773 IC50 = 1700 nM T63966 CY30FL 123752658 IC50 = 62.7 nM T63966 C8KXV1 127025843 IC50 > 1000 nM T63966 CKS28E 127034802 IC50 = 159 nM T63966 CKX40V 127037812 IC50 = 4.9 nM T63966 C70RUP 127038480 IC50 = 9.3 nM T63966 C8TB3R 127041351 IC50 = 3 nM T63966 C40WEH 127041352 IC50 = 7.7 nM T63966 C3WCN8 127041777 IC50 = 4.2 nM T63966 CHK16Q 127045929 IC50 > 1000 nM T63966 CY3J0C 127047591 IC50 > 1000 nM T63966 C5IBZ8 129851326 IC50 = 540 nM T63966 CUO0C5 132156633 IC50 > 10000 nM T63966 CJ04HZ 132585195 IC50 = 159 nM T63966 CERS64 132937256 IC50 > 30000 nM T63966 CYL5V1 134694986 IC50 > 30000 nM T63966 CLCO61 135398510 IC50 = 3 nM T63966 C76JPR 135405015 IC50 = 161 nM T63966 CMVS34 135410282 IC50 = 28 nM T63966 C34FSG 135410286 IC50 = 184 nM T63966 CV8Q7A 135430397 IC50 = 163 nM T63966 C8X5SV 135433815 IC50 = 162 nM T63966 C1M3PW 135458467 IC50 = 10 nM T63966 CS63IO 135476717 IC50 = 34 nM T63966 C9D2FL 135483378 IC50 = 405 nM T63966 CA80OZ 135488014 IC50 = 62 nM T63966 CDCF48 135488027 IC50 = 96 nM T63966 C69FTB 135496141 IC50 = 4300 nM T63966 CG5HY4 135507297 IC50 = 112 nM T63966 CT0NV5 135514617 IC50 = 691 nM T63966 CFPV27 135543821 IC50 = 184 nM T63966 CRCH86 135546221 IC50 > 1950 nM T63966 C65XMQ 135546228 IC50 = 66 nM T63966 CBSV42 135674149 IC50 = 12 nM T63966 C1NTB0 135674153 IC50 = 10 nM T63966 C0PVG7 135819982 IC50 = 1 nM T63966 CQ92DH 135819983 IC50 = 21 nM T63966 C9ZI5J 135820026 IC50 = 28 nM T63966 C9LG3C 135820141 IC50 = 8 nM T63966 CWI61Y 135820280 IC50 = 63 nM T63966 C53LFX 135820297 IC50 = 3 nM T63966 CM2AO1 135820333 IC50 = 50 nM T63966 C5BI9T 135820431 IC50 = 11 nM T63966 CYHV16 135820505 IC50 > 3000 nM T63966 CXJ19P 135839366 IC50 = 602 nM T63966 C0QH5E 135839368 IC50 = 37 nM T63966 C01OLI 135839369 IC50 = 691 nM T63966 CP1H7K 135839370 IC50 = 3940 nM T63966 C2PIQ9 135839371 IC50 = 74 nM T63966 CK6H2P 135839372 IC50 = 132 nM T63966 CXM75Z 135985610 IC50 = 201 nM T63966 C23SGN 136038438 IC50 = 150 nM T63966 CS91JC 136038439 IC50 = 2 nM T63966 C5DVE4 136038477 IC50 > 3000 nM T63966 CAG34B 136038492 IC50 = 170 nM T63966 C7Q1KT 136038570 IC50 > 3000 nM T63966 C9SL4U 136038593 IC50 = 4 nM T63966 CAXJ50 136043793 IC50 = 28 nM T63966 CF12ME 136043801 IC50 = 15 nM T63966 CE4Y0B 136043806 IC50 = 96 nM T63966 C7JF8X 136043808 IC50 = 48 nM T63966 CTAY92 136043832 IC50 = 44 nM T63966 CU05YS 136118622 IC50 = 374 nM T63966 CN49OS 136118623 IC50 = 381 nM T63966 C39CXW 136118624 IC50 = 4322 nM T63966 CR48NF 136118625 IC50 = 24400 nM T63966 CD5M9T 136118626 IC50 = 1950 nM T63966 CW27AO 136118641 IC50 = 1950 nM T63966 CZHA29 136118700 IC50 = 618 nM T63966 CFD03R 136118701 IC50 = 681 nM T63966 C3SIK1 136118702 IC50 = 599 nM T63966 C4LC2Q 136118703 IC50 = 2308 nM T63966 CX39CA 136118704 IC50 = 522 nM T63966 C3PI2X 136118707 IC50 = 2551 nM T63966 C2OAK8 136118708 IC50 = 1796 nM T63966 C6PUG0 136118709 IC50 = 24000 nM T63966 CH1E7I 136118710 IC50 = 24400 nM T63966 C0RBJ7 136118711 IC50 = 984 nM T63966 C4V8HY 136118712 IC50 = 10543 nM T63966 CZ4AF8 136118717 IC50 = 371 nM T63966 CMP78A 136118718 IC50 = 118 nM T63966 CN8RB4 136118719 IC50 = 4544 nM T63966 CIUJ95 136118720 IC50 = 4880 nM T63966 C2BIZ5 136118721 IC50 = 39 nM T63966 C5YL7I 136118722 IC50 = 582 nM T63966 CZQ5P1 136118733 IC50 = 20716 nM T63966 CMP4R8 136118734 IC50 = 45 nM T63966 C7E6XJ 136118735 IC50 = 473 nM T63966 CCX81R 136118736 IC50 = 77 nM T63966 C29ZXF 136118737 IC50 = 377 nM T63966 CDT7E4 136211077 IC50 > 100 nM T63966 CCM42D 137249694 IC50 = 99.2 nM T63966 CXC69T 137321158 IC50 = 76 nM T63966 C25ERN 137631967 IC50 > 10 nM T63966 CI1E8V 137634241 IC50 = 9130 nM T63966 CZ4XO5 137635974 IC50 = 50400 nM T63966 C06JRX 137637094 IC50 = 1 nM T63966 C3KV9G 137639956 IC50 = 75100 nM T63966 CRMB09 137643789 IC50 = 157400 nM T63966 CXK62C 137644697 IC50 = 271100 nM T63966 C3SJ8L 137645340 IC50 = 129500 nM T63966 CJ1IN0 137650005 IC50 = 56000 nM T63966 C1DK0P 137651391 IC50 > 10 nM T63966 CN3LV5 137653006 IC50 = 10400 nM T63966 CV5H3Z 137657932 IC50 > 10 nM T63966 CQMB10 137658515 IC50 = 3493 nM T63966 CIWG23 138393067 IC50 = 22 nM T63966 CSRI06 138547901 IC50 > 1000 nM T63966 CUXO19 138617501 IC50 > 1000 nM T63966 CI1D9F 139600335 IC50 = 22 nM T63966 CB3Z1W 145949428 IC50 = 25 nM T63966 C5VSC7 145956704 IC50 = 23 nM T63966 CY54UC 145957309 IC50 = 220.19 nM T63966 CTUF34 145966712 IC50 = 35 nM T63966 C31JEU 145990213 IC50 = 1900 nM T63966 C9P2FS 145992282 IC50 = 2500 nM T63966 C2MD1Q 155513187 IC50 > 10000 nM T63966 C86HPW 155518524 IC50 = 43000 nM T63966 CXFH76 155523422 IC50 = 845 nM T63966 C8H1CZ 155536201 IC50 = 2100 nM T63966 C7SF2C 155547229 IC50 = 418 nM T63966 CW34RN 155549665 IC50 = 5.5 nM T63966 CYO3B0 155554258 IC50 = 9.6 nM T63966 CQ1N7J 155564622 IC50 = 1255 nM T63966 CX8I9K 155567999 IC50 = 7.1 nM T63966 C6MEO1 155568894 IC50 = 196000 nM T63966 C94IJB 10367131 IC50 = 11 nM T63966 CI8LX0 57976125 IC50 = 29 nM T63966 D00ERW 44444843 Ki > 440 nM T63966 D00HVA 11624601 Ki > 440 nM T63966 D02BXJ 46864270 IC50 = 5.2 nM T63966 D02MFX 44428818 IC50 = 19300 nM T63966 D04ZWF 53396311 IC50 > 5000 nM T63966 D07ADX 54764565 IC50 = 39 nM T63966 D07IHM 9823787 IC50 > 10000 nM T63966 D07OXC 11650194 IC50 > 1000 nM T63966 D07SRX 9797919 IC50 = 180 nM T63966 D09PLJ 11499583 IC50 > 1250 nM T63966 D09QBA 23378546 IC50 > 10000 nM T63966 D0C2GE 67161540 IC50 = 7 nM T63966 D0C6KI 5329006 IC50 = 2000 nM T63966 D0CM6T 11314340 Ki > 2200 nM T63966 D0EE6A 6398883 IC50 = 130 nM T63966 D0IR6U 5494425 IC50 = 1520 nM T63966 D0K7FA 46831062 IC50 = 25000 nM T63966 D0KH5T 5687 IC50 = 200 nM T63966 D0M4QA 56935577 IC50 = 1.3 nM T63966 D0Q3KS 9957049 IC50 > 5000 nM T63966 D0Q3NG 11715520 Ki > 440 nM T63966 D0Q4EQ 16742063 IC50 = 4420 nM T63966 D0R0XY 23630507 IC50 = 39900 nM T63966 D0R2WK 16038120 EC50 = 872 nM T63966 D0S7IE 11658882 Ki > 440 nM T63966 D0XC6G 135464491 IC50 = 720 nM T63966 D0Y0BK 11524144 IC50 = 11 nM T63966 D0Z7TM 22273644 IC50 = 268 nM T11808 CS12YK 80289 IC50 = 501187.23 nM T11808 CJ5E1V 119072 Ki = 22900 nM T11808 CO5Y7H 725447 Ki = 112000 nM T11808 CPJ28H 828532 IC50 = 140 nM T11808 CJ1GN3 869194 Ki = 107000 nM T11808 CBFT53 975107 IC50 = 1300 nM T11808 C97ZIP 2262135 Ki = 100000 nM T11808 C74DMH 2262990 Ki = 95000 nM T11808 CQPJ74 2938648 IC50 = 990 nM T11808 C6WU4N 5000438 IC50 = 1140 nM T11808 CV98LI 5473234 Ki = 22900 nM T11808 CI69XU 5739522 Ki = 121000 nM T11808 C52VYB 8072734 IC50 > 30000 nM T11808 CG51HY 10695695 IC50 = 112 nM T11808 C3TOL6 23106311 IC50 = 19952.62 nM T11808 CLG98H 25258454 Ki = 70700 nM T11808 CAF89H 25400592 IC50 = 200 nM T11808 CS9TK6 38335241 IC50 = 1100 nM T11808 CL0U1A 44303806 IC50 = 7943.28 nM T11808 CW5V7Y 44559839 IC50 = 12500 nM T11808 C0Y7GN 53736009 IC50 = 15848.93 nM T11808 C57MTC 70686944 Ki = 357100 nM T11808 C3I4BR 70691122 Ki = 70400 nM T11808 C15UJW 70693241 Ki = 70700 nM T11808 CQ51CP 70695325 Ki = 200000 nM T11808 C8B5HU 70695326 Ki = 71900 nM T11808 C78DJQ 71711730 IC50 < 10000 nM T11808 CK1OU9 76285535 Ki = 400 nM T11808 CGO0Z1 76310236 IC50 = 156900 nM T11808 CWM9B8 76310252 IC50 = 376600 nM T11808 CNA8X2 76313929 Ki = 2400 nM T11808 C2T1NM 76317472 IC50 = 520700 nM T11808 C0UV9P 76317473 Ki = 26600 nM T11808 CF8PS2 76317474 Ki = 28200 nM T11808 COS46N 76317475 IC50 = 157400 nM T11808 CMW2Z5 76321196 Ki = 1700 nM T11808 CX3W6J 76324824 IC50 = 479800 nM T11808 CB5G6Y 76328377 IC50 = 222900 nM T11808 C49CQJ 76328378 Ki = 2400 nM T11808 CGX1W8 76328379 IC50 = 356600 nM T11808 CY25WA 76328380 Ki = 700 nM T11808 CAEK65 76332053 IC50 = 53900 nM T11808 CZ7TH6 76335659 IC50 = 320600 nM T11808 CN8O7Z 76335660 Ki = 3400 nM T11808 CKC21D 76335671 Ki = 300 nM T11808 CY3O9X 76335672 Ki = 600 nM T11808 CKJN32 122164799 IC50 > 30000 nM T11808 C6RDX4 122192767 Ki = 2.1 nM T11808 CY0K9V 122192770 Ki = 5.2 nM T11808 CDCG19 122192781 Ki = 362 nM T11808 CD5SN7 122192782 Ki > 50000 nM T11808 C4JC0Q 127034134 IC50 = 122 nM T11808 C57LJQ 127034403 IC50 = 115 nM T11808 CW9NJ0 134415778 IC50 = 130 nM T11808 CCY58U 137210069 Ki = 22900 nM T11808 COJ20R 137322719 IC50 = 501.19 nM T11808 CPY9O5 137348758 IC50 > 30000 nM T11808 CDQ62V 137637214 Ki = 50000 nM T11808 C2K8JV 137639385 Ki = 800 nM T11808 CNX46H 137654508 Ki > 50000 nM T11808 CUZ35A 138115400 IC50 = 79.43 nM T11808 CZO2X5 145961109 IC50 > 30000 nM T11808 C7X5MP 145961398 IC50 > 30000 nM T11808 CT2PO1 145961920 IC50 > 30000 nM T11808 C5U0VI 145968421 IC50 > 30000 nM T11808 CAG81E 155511419 IC50 = 39.81 nM T11808 CZR36C 155511554 IC50 = 6.31 nM T11808 CV5F4A 155511614 IC50 = 3981.07 nM T11808 CEJC57 155512056 IC50 = 3600 nM T11808 C1GYM7 155513506 IC50 = 2511.89 nM T11808 C4IZX3 155514387 IC50 = 39810.72 nM T11808 CMY9P0 155514527 IC50 = 6309.57 nM T11808 CW2X7K 155514934 IC50 = 199.53 nM T11808 CD19EV 155517012 IC50 = 17000 nM T11808 C0OY1S 155518519 IC50 = 199526.23 nM T11808 C6NX4K 155519661 IC50 = 0.5012 nM T11808 C4MS1B 155519676 IC50 = 10 nM T11808 CT4L1S 155520177 IC50 = 794.33 nM T11808 CG2WM9 155520998 IC50 = 10000 nM T11808 C41TFK 155521732 IC50 = 10000 nM T11808 C49DMZ 155522189 IC50 = 15848.93 nM T11808 CLM04O 155522595 IC50 = 79.43 nM T11808 CIH95K 155523037 IC50 = 12589.25 nM T11808 C2KM7D 155524369 IC50 = 10000 nM T11808 CRC6L7 155524551 Ki = 3.7 nM T11808 C0MUB5 155525046 IC50 = 1584.89 nM T11808 CSPB43 155525076 IC50 = 2511.89 nM T11808 C6L1WU 155525184 Ki = 143 nM T11808 COT61Y 155526156 IC50 = 6309.57 nM T11808 CIPV21 155526440 IC50 = 63.1 nM T11808 CXBR96 155526691 IC50 = 6309.57 nM T11808 CN3BH5 155527998 IC50 = 25.12 nM T11808 CHYW65 155528639 IC50 = 1.259 nM T11808 CKW0N3 155528746 IC50 = 25118.86 nM T11808 CD7O2G 155530095 IC50 = 7.943 nM T11808 C42LDK 155530603 IC50 = 6309.57 nM T11808 C9QA5T 155530999 IC50 = 7000 nM T11808 C35QWO 155531023 IC50 < 0.7943 nM T11808 CENG47 155531694 IC50 = 79.43 nM T11808 CDT7A9 155531797 Ki = 0.34 nM T11808 CIH96R 155532277 IC50 = 251.19 nM T11808 C9CH2J 155532630 IC50 = 10000 nM T11808 CG03WZ 155533183 IC50 = 794.33 nM T11808 CC2TH3 155534011 IC50 = 19952.62 nM T11808 C3R0PV 155535171 IC50 = 79.43 nM T11808 C12HON 155536142 IC50 = 12.59 nM T11808 C7RBN1 155536236 IC50 = 158.49 nM T11808 CUW43P 155537713 IC50 = 1800 nM T11808 CMG5X7 155538944 Ki = 8.9 nM T11808 CVCN73 155539549 IC50 = 398107.17 nM T11808 CR3HF2 155539807 IC50 = 6309.57 nM T11808 CYQ5N7 155540505 IC50 = 125892.54 nM T11808 C0IXU7 155540672 IC50 = 2511.89 nM T11808 C8N9QK 155540725 IC50 = 4900 nM T11808 CY6DK3 155540964 IC50 = 5.012 nM T11808 C2PL7Y 155541127 IC50 = 125.89 nM T11808 C97IBT 155542437 IC50 = 39810.72 nM T11808 CHYZ70 155544016 IC50 = 5011.87 nM T11808 CX86UZ 155545827 IC50 = 12000 nM T11808 CU52QS 155545897 Ki > 10000 nM T11808 CH2S6R 155546346 Ki > 10000 nM T11808 CX9A5M 155547612 IC50 < 10 nM T11808 C5MB9R 155547962 IC50 = 7.943 nM T11808 CG8F4S 155548359 IC50 = 12589.25 nM T11808 CLFB25 155548371 IC50 = 7.943 nM T11808 C75CKY 155550727 IC50 = 12589.25 nM T11808 COM52R 155551892 IC50 = 6.31 nM T11808 CJ3FI5 155553630 IC50 = 25.12 nM T11808 CMV2T0 155553751 IC50 = 79.43 nM T11808 C5BH7C 155553819 IC50 = 10000 nM T11808 CT9ZK6 155554786 IC50 = 14000 nM T11808 C9BKN7 155554975 IC50 = 316.23 nM T11808 CVGQ48 155555178 Ki = 0.73 nM T11808 CSW48V 155557718 IC50 < 0.3162 nM T11808 CFZ8Y9 155557932 IC50 = 3981.07 nM T11808 CNOI61 155558524 IC50 = 31622.78 nM T11808 CNZ1K5 155559920 Ki > 10000 nM T11808 C6D8KL 155560348 IC50 = 12589.25 nM T11808 C4CTA0 155562690 IC50 = 8000 nM T11808 CZI5S1 155563470 IC50 = 50118.72 nM T11808 C6N0LM 155564043 Ki = 2.4 nM T11808 CM8XB1 155565537 IC50 = 3.981 nM T11808 C8N3SP 155566632 IC50 = 1000 nM T11808 CAK16X 155566796 IC50 = 158489.32 nM T11808 CN6BS0 155567190 IC50 = 31.62 nM T11808 CIU2C9 155568927 IC50 = 100 nM T11808 D00LOL 970375 IC50 = 270 nM T11808 D0Y5IQ 44255320 IC50 = 10000 nM T97016 D0E3TC 44259 IC50 = 1.21 nM T97016 D03BNU 59604787 IC50 > 10000 nM T97016 C3VRO9 44557921 IC50 > 10000 nM T97016 CV63UL 67240318 IC50 > 10000 nM T97016 C3TS2A 132968992 IC50 = 490 nM T97016 C2MD1Q 155513187 IC50 > 10000 nM T97016 D00ERW 44444843 Ki > 9334 nM T97016 D08HFG 24809764 IC50 = 420 nM T17980 D03ZBT 11626560 IC50 > 10000 nM T17980 D0E6XR 3062316 IC50 < 0.5 nM T17980 D0OB0F 5328940 IC50 = 410 nM T17980 D0T7OW 681 IC50 > 100000 nM T17980 D00UZR 5330286 IC50 > 10000 nM T17980 D03AND 11656518 IC50 > 10000 nM T17980 D03LWG 53235510 IC50 = 1900 nM T17980 D04AHQ 71721540 IC50 = 91 nM T17980 D07EHV 44814409 IC50 > 10000 nM T17980 D08HOM 46207586 IC50 = 110 nM T17980 D0E3TC 44259 IC50 = 2 nM T17980 D0L4FS 5280961 IC50 = 58180 nM T17980 D00OWF 5280953 IC50 > 250000 nM T17980 D04FHB 6918852 Ki > 5000 nM T17980 D09HEV 6539952 IC50 = 0.3 nM T17980 D0T3ME 156422 IC50 = 24000 nM T17980 CB1VW3 1400 IC50 = 10 nM T17980 CK1JY9 3106 IC50 > 100000 nM T17980 CJ17AM 4877 IC50 = 600 nM T17980 CBPM40 4878 IC50 = 10 nM T17980 CF6WU5 125246 IC50 = 50000 nM T17980 CIE63B 446044 IC50 > 200000 nM T17980 CY13FW 644243 IC50 = 1 nM T17980 C9U7NK 1128774 IC50 = 68540 nM T17980 C4C0KQ 1430509 Ki = 2100 nM T17980 CM5VN6 4600415 IC50 = 38670 nM T17980 C76ORW 5328887 IC50 > 10000 nM T17980 CS6L2C 5328911 IC50 > 10000 nM T17980 C16ECF 5328912 IC50 > 10000 nM T17980 C23VOL 5328913 IC50 = 3200 nM T17980 C8LGK5 5328914 IC50 = 2900 nM T17980 CH83QU 5328915 IC50 = 4500 nM T17980 CM98RH 5330099 IC50 = 580 nM T17980 CUEZ35 5330437 IC50 = 420 nM T17980 C94GRU 5330453 IC50 = 1170 nM T17980 CH2JS0 5330459 IC50 = 830 nM T17980 CPQV76 5353678 IC50 > 100000 nM T17980 CP0XI6 6603792 IC50 = 126 nM T17980 CI80BK 9803350 IC50 = 300 nM T17980 C6QBF8 9823235 Ki = 100 nM T17980 CRC65X 9863786 IC50 > 10000 nM T17980 C2TC1L 9910609 IC50 = 322 nM T17980 CYW49X 9927718 IC50 = 71 nM T17980 CRK63X 9933645 Ki = 2.4 nM T17980 CWBC91 9992262 IC50 > 100000 nM T17980 C5ZY0I 10050705 IC50 = 10000 nM T17980 CD30IN 10241671 IC50 = 1000 nM T17980 C6DC8Q 10275163 IC50 = 60 nM T17980 C7SFI1 10296883 IC50 = 5500 nM T17980 C5CBF9 10320381 IC50 = 50 nM T17980 CPS79C 10402283 IC50 = 20 ug.mL-1 T17980 CLAX64 10413508 IC50 = 1200 nM T17980 CC2L5P 10467257 IC50 = 10000 nM T17980 CJ5M1D 10482445 IC50 = 400 nM T17980 CF2GE5 11222252 Ki = 3500 nM T17980 CVOW82 11238420 IC50 = 35100 nM T17980 CBOP58 11293798 Ki > 10000 nM T17980 C26BZX 11362471 Ki > 10000 nM T17980 CWXB93 11397177 Ki > 10000 nM T17980 C64IGY 11448608 Ki > 5000 nM T17980 CK3M0T 11495270 IC50 = 11800 nM T17980 CTG83F 11539329 Ki > 810 nM T17980 CACS26 11561968 Ki > 2000 nM T17980 CO9KP5 11583459 IC50 > 10000 nM T17980 C3VUO7 11588815 IC50 > 12500 nM T17980 CA2KX0 11590078 IC50 > 50000 nM T17980 CMIL86 11590363 Ki > 810 nM T17980 C9T6SC 11640926 Ki > 810 nM T17980 CU0E8O 11690457 Ki > 2000 nM T17980 CB0AP2 11705863 Ki > 2000 nM T17980 CZY05V 11719421 IC50 = 23 nM T17980 CE0KI4 11753519 IC50 = 25900 nM T17980 CP7AH3 11755812 IC50 = 50000 nM T17980 CT47ES 12728243 IC50 > 100000 nM T17980 CW48TD 15159374 IC50 = 900 nM T17980 C3SYC4 15159375 IC50 = 19 nM T17980 C7V5WC 15159376 IC50 = 9700 nM T17980 CQ49GK 15159377 IC50 = 340 nM T17980 C3FH4K 15159378 IC50 = 32 nM T17980 C0KQD6 15159379 IC50 = 670 nM T17980 C95SKG 15159380 IC50 = 150 nM T17980 CJKX79 15159381 IC50 = 1400 nM T17980 C2DKN0 15159382 IC50 = 540 nM T17980 C3YRU7 15295578 IC50 > 50000 nM T17980 CFPW41 16007116 IC50 > 810 nM T17980 C09OWB 16015442 IC50 = 600 nM T17980 CFKE48 16064750 IC50 = 220 nM T17980 CGC34R 16118737 IC50 = 3 nM T17980 C5VPH9 16129448 IC50 = 1030 nM T17980 CP3HS4 16220354 IC50 = 27300 nM T17980 CHZ75U 16663089 IC50 = 100 nM T17980 CDZ31W 16747696 IC50 > 50000 nM T17980 CJA0D6 18451024 IC50 = 26200 nM T17980 C6FQB7 18451036 IC50 = 44100 nM T17980 CEU1O0 20817327 IC50 > 50000 nM T17980 CK1TF6 20817330 IC50 > 50000 nM T17980 C6AN8E 20817403 IC50 = 1070 nM T17980 C56HRP 20817416 IC50 > 50000 nM T17980 CXCF38 20817425 IC50 > 50000 nM T17980 CGX61W 22041319 IC50 = 5 nM T17980 CQ2XW6 22346679 IC50 >= 50000 nM T17980 CZRT79 22346947 IC50 > 50000 nM T17980 CG12OL 23518511 IC50 = 500 nM T17980 CE7K3W 23532567 IC50 > 10000 nM T17980 CA3I4T 24753787 IC50 > 50000 nM T17980 C2UOE0 24766030 IC50 = 25 nM T17980 CCP2M3 24822704 IC50 > 50000 nM T17980 CS3Q8B 24995659 IC50 > 2000 nM T17980 CX3F4U 25195515 IC50 = 58200 nM T17980 CLFM35 25206064 IC50 > 50000 nM T17980 CI9DK5 42628614 IC50 = 1100 nM T17980 CLW80F 44160269 IC50 = 1700 nM T17980 CK73NR 44219749 IC50 > 50000 nM T17980 CG1C9E 44269392 IC50 > 250000 nM T17980 CAT6W7 44269404 IC50 > 250000 nM T17980 C4SA3Y 44269518 IC50 > 250000 nM T17980 CRH2T3 44270586 IC50 = 50000 nM T17980 C5UPO8 44270599 IC50 = 10000 nM T17980 CX5E7N 44270619 IC50 > 100000 nM T17980 CQ97UV 44270641 IC50 = 10000 nM T17980 C8R3UZ 44270657 IC50 = 10000 nM T17980 CH3J2E 44299176 IC50 = 400 nM T17980 C27GVO 44299203 IC50 = 1400 nM T17980 CY6WC0 44299236 IC50 = 400 nM T17980 C3RG0C 44299304 IC50 = 600 nM T17980 CJM26I 44299321 IC50 = 200 nM T17980 C9UGL3 44299325 IC50 = 800 nM T17980 CJEZ96 44299338 IC50 = 400 nM T17980 C8XGN5 44299339 IC50 = 200 nM T17980 CNH34G 44299354 IC50 = 100 nM T17980 C82MSD 44299360 IC50 = 700 nM T17980 CEZF96 44303555 IC50 = 630 nM T17980 CO81DL 44318069 IC50 = 3 ug.mL-1 T17980 C4KS5N 44320732 IC50 = 4 nM T17980 CC6YI7 44320769 Ki = 1.1 nM T17980 CXM61A 44321260 Ki = 8.8 nM T17980 C2FST3 44324647 IC50 = 100 nM T17980 CI8YR0 44324649 IC50 = 11000 nM T17980 C7JYP4 44324728 IC50 = 45000 nM T17980 CY69SU 44324769 IC50 = 33000 nM T17980 C7PBJ8 44405918 IC50 > 50000 nM T17980 C0GR5F 44405919 IC50 = 32500 nM T17980 CO5WU8 44405977 IC50 > 50000 nM T17980 C9LX5Q 44406001 IC50 > 50000 nM T17980 CQ4U7T 44406037 IC50 > 50000 nM T17980 CEVF48 44406058 IC50 > 50000 nM T17980 CF46WP 44406078 IC50 > 50000 nM T17980 CUQ6R8 44406079 IC50 = 13600 nM T17980 CG2W4V 44406138 IC50 > 50000 nM T17980 CGV37F 44440254 IC50 = 13681 nM T17980 C5JUV3 44440256 IC50 > 50000 nM T17980 CFB56S 44440259 IC50 = 22986 nM T17980 CEW9G2 44440261 IC50 > 50000 nM T17980 C9Z8XJ 44460238 IC50 > 20 ug.mL-1 T17980 CV1Q0D 44460258 IC50 > 20 ug.mL-1 T17980 C3VRO9 44557921 IC50 > 10000 nM T17980 CJY8S0 44570884 IC50 > 5000 nM T17980 CCL85F 44575073 IC50 > 50000 nM T17980 CJX06P 44575126 IC50 > 50000 nM T17980 CE8FC7 44575127 IC50 = 15300 nM T17980 C28QLM 44605035 IC50 > 50000 nM T17980 C75XHS 44605037 IC50 > 50000 nM T17980 CC95PQ 45375865 IC50 = 140 nM T17980 CEOQ27 45375866 IC50 > 50000 nM T17980 C96BNW 46179972 IC50 = 5 nM T17980 CY3HW5 46224684 IC50 > 10000 nM T17980 CYT37A 46232443 IC50 > 50000 nM T17980 C48ZVW 46232555 IC50 = 28000 nM T17980 CS9B1U 46232556 IC50 = 25000 nM T17980 CO3P0J 46866604 IC50 < 50000 nM T17980 CLS29B 46872626 IC50 > 10000 nM T17980 CJOM49 46880136 IC50 = 1940 nM T17980 C2O8RZ 46886323 IC50 > 1000 nM T17980 CL0O4U 46911726 Ki = 28 nM T17980 C0B6KG 46976768 Ki = 2250 nM T17980 CHSF07 49806372 IC50 > 1000 nM T17980 CTZ9U6 50913410 Ki = 1150 nM T17980 CEQN27 52936621 Ki > 1000 nM T17980 C9UH8Q 52951545 Ki = 8150 nM T17980 C2MVU5 52951547 Ki = 15500 nM T17980 CBI6V7 52951665 Ki = 7500 nM T17980 C1KYR9 53326941 IC50 = 22000 nM T17980 CD4H3S 53354074 Ki > 1000 nM T17980 C8NA4L 53384644 IC50 > 30000 nM T17980 C8AB1J 54759606 Ki = 1800 nM T17980 C9DX3J 56649281 IC50 = 11.09 nM T17980 CR16SD 56947170 IC50 = 750 nM T17980 CPHX64 57325478 IC50 > 50000 nM T17980 CQ9BW4 57325479 IC50 > 50000 nM T17980 CE1A9V 57394653 IC50 = 892 nM T17980 CVK0G4 58056356 IC50 > 50000 nM T17980 C1EVX0 58063117 IC50 = 4970 nM T17980 CWXC70 58180596 IC50 = 10 nM T17980 CLH49Z 59790029 IC50 = 2 nM T17980 C1MR8Q 60097495 IC50 > 10000 nM T17980 C9QRX3 60098131 IC50 = 40 nM T17980 CE49GC 67098566 Ki = 80 nM T17980 C37NKO 67129970 IC50 = 5330 nM T17980 CK80LJ 67130050 IC50 = 5960 nM T17980 CV63UL 67240318 IC50 > 10000 nM T17980 C7GRV2 68755406 IC50 = 1510 nM T17980 CAIO65 68796885 IC50 = 131 nM T17980 C1IEJ2 70789254 IC50 = 158000 nM T17980 C8T7ZP 70789255 IC50 = 26000 nM T17980 COU73Y 71226944 IC50 = 188 nM T17980 C40JOZ 71235465 IC50 = 571 nM T17980 CKT60L 71455860 Ki = 328 nM T17980 CDJY72 71568837 IC50 = 2800 nM T17980 C8CAG7 71578921 IC50 > 10000 nM T17980 CSUZ81 73356106 IC50 > 200000 nM T17980 CPG3A5 86302574 IC50 = 11161 nM T17980 CQCX41 118737057 IC50 = 5 nM T17980 CKBP72 121231408 IC50 = 2.1 nM T17980 CJPL50 121316007 Ki = 16000 nM T17980 C3OJ5F 121316011 Ki = 95 nM T17980 C81QZH 121316014 Ki = 900 nM T17980 C8I9MR 121316037 Ki = 10000 nM T17980 CZ2SV7 121316042 Ki = 3350 nM T17980 CI52KS 121316045 Ki = 995 nM T17980 C3JK0M 121316054 Ki = 13000 nM T17980 C4J0AI 121316056 Ki = 10000 nM T17980 CMP3X7 121316059 Ki = 1625 nM T17980 C7QLK6 121316061 Ki = 10000 nM T17980 CDSV38 121316062 Ki = 70 nM T17980 C87ZID 121316067 Ki = 12500 nM T17980 CMB2W9 121316084 Ki = 360 nM T17980 CLIM03 121316090 Ki = 870 nM T17980 CD6S3B 121316093 Ki = 1485 nM T17980 CA41IM 121316143 Ki = 1400 nM T17980 C81IFQ 122163152 IC50 > 100000 nM T17980 C4X7SD 122192466 IC50 > 10000 nM T17980 CD67LU 122705248 IC50 = 38 nM T17980 CX63VW 122705258 IC50 = 1964 nM T17980 C76IKM 122705261 IC50 = 1226 nM T17980 C8ALO2 124088839 IC50 = 913 nM T17980 CG8DA9 127045861 IC50 > 100000 nM T17980 CC4ND8 127046862 IC50 > 100000 nM T17980 CO25WH 127052538 IC50 = 311 nM T17980 C8F0DQ 129909860 IC50 = 45 nM T17980 C2KFH7 135398497 Ki > 2000 nM T17980 CS4OW8 135400873 Ki > 2000 nM T17980 C2DH1R 135412832 IC50 > 20 ug.mL-1 T17980 CFAD48 135611170 Ki > 2000 nM T17980 C5XIE8 136026041 IC50 = 17000 nM T17980 CVIC49 136069671 IC50 = 1300 nM T17980 CPE2B1 136185998 IC50 = 20 ug.mL-1 T17980 CR9XE0 136185999 IC50 > 20 ug.mL-1 T17980 C1I8LC 136186000 IC50 > 20 ug.mL-1 T17980 C40HWO 136186001 IC50 > 20 ug.mL-1 T17980 CGP04W 136186009 IC50 > 20 ug.mL-1 T17980 CS5QE7 136186010 IC50 > 20 ug.mL-1 T17980 CXC69T 137321158 IC50 = 187 nM T17980 CZOD53 137633880 IC50 = 894 nM T17980 CI1E8V 137634241 IC50 = 201 nM T17980 C7BJY5 137636807 IC50 = 248 nM T17980 C07CQL 137637848 IC50 = 30800 nM T17980 CQTF50 137641213 IC50 = 57100 nM T17980 C36KUM 137642749 IC50 = 76000 nM T17980 C7KQH8 137644946 IC50 = 43200 nM T17980 CO89DX 137649100 IC50 = 105 nM T17980 CINE03 137652514 IC50 = 1904 nM T17980 C28QUP 137652864 IC50 = 429.8 nM T17980 C71HKP 137655481 IC50 = 88600 nM T17980 C0YP9H 137657483 IC50 = 62000 nM T17980 C1XW3M 137659733 IC50 = 70400 nM T17980 CRWA29 139030520 IC50 = 165.2 nM T17980 C2MD1Q 155513187 IC50 > 10000 nM T17980 C3NA2I 155519537 IC50 = 232 nM T17980 CY5MR2 155522337 Ki = 120 nM T17980 C3V4LG 155538413 IC50 = 191 nM T17980 D00ERW 44444843 Ki > 809 nM T17980 D00HVA 11624601 Ki > 810 nM T17980 D01VFR 4708 IC50 = 420 nM T17980 D01YWE 25207521 IC50 > 50000 nM T17980 D03AER 9549185 IC50 > 50000 nM T17980 D03OKV 9844320 IC50 > 5 nM T17980 D04PEI 11467730 IC50 = 1100 nM T17980 D05PTT 5281792 IC50 = 3600 nM T17980 D06HVH 54613583 IC50 > 10000 nM T17980 D06WGX 9549184 IC50 = 44100 nM T17980 D07IHM 9823787 IC50 = 1190 nM T17980 D08RZB 11153014 IC50 = 1 nM T17980 D09QBA 23378546 IC50 = 3400 nM T17980 D09XIL 11396738 IC50 = 466 nM T17980 D0AH5T 5626 IC50 > 100000 nM T17980 D0CE3R 5312137 IC50 = 170 nM T17980 D0GT8N 5154691 IC50 = 1000 nM T17980 D0IR6U 5494425 IC50 = 500 nM T17980 D0N8TQ 10401956 IC50 = 6 nM T17980 D0Q3NG 11715520 Ki > 810 nM T17980 D0S7IE 11658882 Ki > 810 nM T17980 D0YZ7H 9797370 IC50 = 378 nM T12541 D0J5VR 11625818 IC50 > 10000 nM T12541 D01QSO 16654980 IC50 > 25000 nM T12541 D03LWG 53235510 IC50 > 9000 nM T12541 D07EHV 44814409 IC50 > 9100 nM T12541 D08QGT 17755052 IC50 > 10000 nM T12541 D0O6VZ 25254071 IC50 > 10000 nM T12541 C1O4KS 4416330 IC50 = 10000 nM T12541 CIN5F7 4904109 IC50 = 8 nM T12541 C9U2YK 5109813 IC50 = 501.19 nM T12541 CJ9B1R 11220250 IC50 = 4500 nM T12541 CO9C4H 11348293 IC50 = 8290 nM T12541 C8ENV0 15956160 IC50 = 3080 nM T12541 CEYL29 23585510 IC50 = 240 nM T12541 CBL37C 23642173 IC50 = 40 nM T12541 CB79YC 24905143 IC50 = 2600 nM T12541 CN6V8Z 24905145 IC50 = 17 nM T12541 CVDG02 24905150 IC50 = 6370 nM T12541 CWH6C5 24905152 IC50 = 8 nM T12541 C0HE2Q 24905153 IC50 = 99 nM T12541 C7QSC9 24905154 IC50 = 5700 nM T12541 CO9D0K 24905155 IC50 = 3400 nM T12541 C5W9UR 24905157 IC50 = 1700 nM T12541 CC1DA3 24905158 IC50 = 2800 nM T12541 COW79F 24905159 IC50 = 4900 nM T12541 CFPA53 24905160 IC50 = 7200 nM T12541 C2O0JX 24905161 IC50 = 2000 nM T12541 CA72BE 24905162 IC50 = 4900 nM T12541 CQN6X9 24905163 IC50 = 12000 nM T12541 CD4O1F 24905165 IC50 = 14000 nM T12541 CKL48T 24905166 IC50 = 3500 nM T12541 C76VYL 24905167 IC50 = 4400 nM T12541 C7K5PU 24905168 IC50 = 7400 nM T12541 CZ57ID 24905169 IC50 = 8200 nM T12541 C2DHX9 24905170 IC50 = 14000 nM T12541 CSB96E 24905171 IC50 = 100000 nM T12541 CWZ0R2 24905172 IC50 = 9100 nM T12541 CY3B6M 24905175 IC50 = 13000 nM T12541 CW7UA3 24905176 IC50 = 3500 nM T12541 CW1V0H 24905177 IC50 = 3000 nM T12541 CO6Y0L 24905178 IC50 = 3600 nM T12541 C60NQW 24905179 IC50 = 4900 nM T12541 C4MO8B 24905180 IC50 = 2780 nM T12541 COJI47 24905181 IC50 = 4020 nM T12541 CS0B2C 24905182 IC50 = 7390 nM T12541 C1H4BT 24905183 IC50 = 530 nM T12541 C4WHK9 24905184 IC50 = 100000 nM T12541 C7Q4MZ 24905185 IC50 = 13000 nM T12541 CS4IP1 24905186 IC50 = 4090 nM T12541 C69QWO 24905187 IC50 = 100000 nM T12541 C85ANB 24905188 IC50 = 4100 nM T12541 CNHD75 24905189 IC50 = 5100 nM T12541 C9JUO2 24905190 IC50 = 2600 nM T12541 CPR03K 24905191 IC50 = 3500 nM T12541 CTAG19 24905193 IC50 = 9800 nM T12541 C7VJM5 24905194 IC50 = 5000 nM T12541 CEP1L3 24905195 IC50 = 5700 nM T12541 CP68ZD 24905196 IC50 = 8000 nM T12541 C8Z0RJ 24905197 IC50 = 5000 nM T12541 CIF2J5 24905251 IC50 = 9300 nM T12541 CPTE58 24905252 IC50 = 4720 nM T12541 CP50RD 24905280 IC50 = 2500 nM T12541 CG13ZM 24905281 IC50 = 2340 nM T12541 CF0S6X 24905282 IC50 = 5500 nM T12541 C5HBL0 24905284 IC50 = 31000 nM T12541 C2Z5DN 24905285 IC50 = 8800 nM T12541 CL6GH8 24905286 IC50 = 3400 nM T12541 CKYO98 24905287 IC50 = 12000 nM T12541 CRNQ65 24905288 IC50 = 3900 nM T12541 COD7I5 24905289 IC50 = 40000 nM T12541 C4LP7E 24905290 IC50 = 100000 nM T12541 CE9JC2 24905291 IC50 = 100000 nM T12541 C2GI1R 24905292 IC50 = 5600 nM T12541 CHW8C4 24905293 IC50 = 100000 nM T12541 CQF0H1 24905294 IC50 = 100000 nM T12541 CNO7X0 24905295 IC50 = 4600 nM T12541 C5WRG7 24905296 IC50 = 1500 nM T12541 CQ1S0U 24905297 IC50 = 12000 nM T12541 C4UES7 24905298 IC50 = 100000 nM T12541 CMS69P 24905299 IC50 = 100000 nM T12541 CC0U5M 24905300 IC50 = 10000 nM T12541 CW7X6S 24905301 IC50 = 100000 nM T12541 C97IQV 24905302 IC50 = 11500 nM T12541 CSJ47V 24905303 IC50 = 100000 nM T12541 CPN74C 24905304 IC50 = 100000 nM T12541 C5CS3N 24905305 IC50 = 100000 nM T12541 CK4XE9 24905307 IC50 = 100000 nM T12541 CTU6Z3 24905308 IC50 = 100000 nM T12541 C9SQX1 24905309 IC50 = 100000 nM T12541 CM75JP 24905310 IC50 = 100000 nM T12541 C9Q2BJ 24905311 IC50 = 18000 nM T12541 C9VUA1 24905312 IC50 = 41200 nM T12541 CU3RS1 24905313 IC50 = 15000 nM T12541 CYG3H2 24905314 IC50 = 24000 nM T12541 CV5Q7O 24905315 IC50 = 4060 nM T12541 C8SA3O 24905316 IC50 = 7800 nM T12541 CI5MN3 24905317 IC50 = 8800 nM T12541 CJ1P7K 24905318 IC50 = 100000 nM T12541 C1T6YQ 24905319 IC50 = 9020 nM T12541 CAU86X 24905320 IC50 = 2860 nM T12541 C54ISY 24905321 IC50 = 31900 nM T12541 C2GE5I 24905322 IC50 = 14600 nM T12541 C8D6YK 24905323 IC50 = 12400 nM T12541 C5NZH9 24905324 IC50 = 12900 nM T12541 C1S0PC 24905335 IC50 = 9000 nM T12541 C9E8BJ 24905338 IC50 = 2700 nM T12541 CX85AC 24905341 IC50 = 24000 nM T12541 CKZ80E 24905342 IC50 = 3700 nM T12541 CO8SH1 24905343 IC50 = 5900 nM T12541 C7IZL6 24905344 IC50 = 5100 nM T12541 C2IM0O 39733146 IC50 = 1258.93 nM T12541 C3VRO9 44557921 IC50 > 10000 nM T12541 CB37KZ 46894120 IC50 = 10 nM T12541 CR5OZ8 46916382 IC50 = 5 nM T12541 CP2QD0 49784894 IC50 = 5200 nM T12541 C7PER0 49853953 IC50 = 4000 nM T12541 C1LBX3 49854049 IC50 = 65 nM T12541 CAU39Y 49854158 IC50 = 160 nM T12541 CPK6X3 49854360 IC50 = 320 nM T12541 C0ORZ9 49854466 IC50 = 210 nM T12541 CN2V8R 49854681 IC50 = 3200 nM T12541 CJPE20 49855193 IC50 = 250 nM T12541 CY36EH 51003592 IC50 = 1000 nM T12541 CRJ5W8 51358113 IC50 = 18.3 nM T12541 CU1P2L 52940797 IC50 = 25000 nM T12541 CDHJ08 52942235 IC50 = 5500 nM T12541 C1XEV2 52943394 IC50 = 100000 nM T12541 CWPC54 52945348 IC50 = 4200 nM T12541 C4NLX7 52945630 IC50 = 4000 nM T12541 CXD6T8 52945845 IC50 = 9100 nM T12541 C7ZH0D 53308041 IC50 = 3440 nM T12541 C10YUH 53318615 IC50 = 1000 nM T12541 CN92LK 53322732 IC50 = 5000 nM T12541 CT6XL0 57466811 IC50 = 1330 nM T12541 C59YAC 57495353 IC50 > 9100 nM T12541 CJ6R8Q 59251679 IC50 = 2350 nM T12541 CUC7B3 66557964 IC50 > 50000 nM T12541 C1HSE0 67035086 IC50 > 9100 nM T12541 C38RGB 67035556 IC50 > 9100 nM T12541 C25AHY 67984037 IC50 = 3800 nM T12541 C8I7GC 68293638 IC50 > 10000 nM T12541 CQS8G7 70686830 IC50 = 920 nM T12541 CNI98B 71525653 IC50 = 4 nM T12541 CED42M 71572529 IC50 = 114 nM T12541 CS9NU1 71572531 IC50 = 115 nM T12541 CHW47S 71572645 IC50 = 9 nM T12541 C2L8XG 71572646 IC50 = 53 nM T12541 CS2CW5 71572648 IC50 = 216 nM T12541 C3W5XI 71573239 IC50 = 424 nM T12541 CX65CB 71597290 IC50 = 8000 nM T12541 CF7R0Y 71682057 IC50 = 53 nM T12541 C4LO5V 71682058 IC50 = 22 nM T12541 CM78WZ 71682209 IC50 = 53 nM T12541 CMG8N0 71682210 IC50 = 40 nM T12541 CRN3A6 71682211 IC50 = 35 nM T12541 CX48CN 71682212 IC50 = 67 nM T12541 C0EMZ1 71682213 IC50 = 48 nM T12541 CQ53SW 71682214 IC50 = 225 nM T12541 CNX76A 72544842 IC50 = 630.96 nM T12541 CFPW17 73348992 IC50 = 100 nM T12541 C0N3RW 76282073 IC50 = 11 nM T12541 CREB28 76282315 IC50 = 1000 nM T12541 C62GWR 76853139 IC50 = 8 nM T12541 C9I7TY 78319187 IC50 = 1584.89 nM T12541 CV6PI8 87562294 IC50 = 3981.07 nM T12541 C9AHJ5 91668195 IC50 = 4 nM T12541 CK4Y2U 91758319 IC50 = 54 nM T12541 C8T3RI 117653382 IC50 = 316 nM T12541 C5R0JB 117653568 IC50 = 635 nM T12541 C6AS1P 117653653 IC50 = 543 nM T12541 C6UOT8 117653759 IC50 = 8 nM T12541 CMX3U8 118107483 IC50 = 3100 nM T12541 CM93VO 118611725 IC50 = 13 nM T12541 C58XRY 122184465 IC50 = 630.96 nM T12541 C16ALM 122184466 IC50 = 630.96 nM T12541 CIX19J 122184467 IC50 = 316.23 nM T12541 CDZY02 122184468 IC50 = 3162.28 nM T12541 CTH70U 122184469 IC50 = 1258.93 nM T12541 C9ZXR7 122184470 IC50 = 1000 nM T12541 CNJ9Z4 122184471 IC50 = 1584.89 nM T12541 CMCP83 122184472 IC50 = 794.33 nM T12541 CS41EG 122184473 IC50 = 501.19 nM T12541 CZ36GL 122184474 IC50 = 1584.89 nM T12541 CU4ZT6 122184475 IC50 = 7943.28 nM T12541 C3H9PR 122184476 IC50 = 501.19 nM T12541 CU40TW 122184477 IC50 = 1000 nM T12541 C8IK9C 122184478 IC50 = 2511.89 nM T12541 CAMD31 122184479 IC50 = 39810.72 nM T12541 C1F9RK 122184480 IC50 = 1000 nM T12541 C7XW1K 122184481 IC50 = 2511.89 nM T12541 CRUX54 122184482 IC50 = 6309.57 nM T12541 CQ7W0P 122184526 IC50 = 6309.57 nM T12541 CA5YB2 122184529 IC50 = 1258.93 nM T12541 C64YPH 122184530 IC50 = 1000 nM T12541 C4AGX5 122184531 IC50 = 1584.89 nM T12541 CQL4K5 122184532 IC50 = 1995.26 nM T12541 CRKV74 122184533 IC50 = 2511.89 nM T12541 CX14YD 122184534 IC50 = 1995.26 nM T12541 CM6A4S 122184535 IC50 = 1995.26 nM T12541 CF86YS 122184536 IC50 = 794.33 nM T12541 CH08SN 122184537 IC50 = 316.23 nM T12541 CYRH97 122184538 IC50 = 316.23 nM T12541 CD4W0Z 122184539 IC50 = 10000 nM T12541 CH8Y3Q 122184540 IC50 = 398.11 nM T12541 CDA85R 122184541 IC50 = 316.23 nM T12541 CF36XJ 122184542 IC50 = 2511.89 nM T12541 CQ6O7H 122184543 IC50 = 630.96 nM T12541 CS4MN0 122184544 IC50 = 251.19 nM T12541 CV95OM 122443833 IC50 = 8795 nM T12541 C19RPD 122443864 IC50 = 2583 nM T12541 C0Q7EK 122443905 IC50 = 85 nM T12541 CAB83Y 122443909 IC50 = 275 nM T12541 CWR61Q 122443951 IC50 = 18 nM T12541 CC2EZ8 122443959 IC50 = 20 nM T12541 C0KD5Q 122443986 IC50 = 1500 nM T12541 CU61IM 122444026 IC50 = 6138 nM T12541 CIT28L 122444047 IC50 = 1764 nM T12541 C2WLN5 122444097 IC50 = 331 nM T12541 CEO76N 123131772 IC50 = 0.98 nM T12541 CQP8L7 123131773 IC50 = 14.9 nM T12541 C2OP5X 123131774 IC50 = 26.9 nM T12541 C16HAI 123131775 IC50 = 22 nM T12541 C8MSY6 134132647 IC50 = 7.23 nM T12541 C4MJ7A 134133351 IC50 = 56 nM T12541 CC68TF 134135057 IC50 = 33.7 nM T12541 C3EVJ9 134136768 IC50 = 19.9 nM T12541 C1DZO4 134137055 IC50 = 17.6 nM T12541 C57ECB 134137863 IC50 = 17.2 nM T12541 C8NWS3 134137978 IC50 = 2.4 nM T12541 CE5TU2 134138026 IC50 = 74.6 nM T12541 CA7Z4G 134138094 IC50 = 134.8 nM T12541 C8UZP7 134139703 IC50 = 43.8 nM T12541 CI5S8B 134140256 IC50 = 6.2 nM T12541 COA46T 134141075 IC50 = 145.4 nM T12541 COZ0C6 134141276 IC50 = 27.3 nM T12541 CC14UO 134142679 IC50 = 26.4 nM T12541 C0IH3R 134145381 IC50 = 444.1 nM T12541 CZQ20R 134146889 IC50 = 146.9 nM T12541 CYM69S 134146987 IC50 = 19.1 nM T12541 C2KU0W 134147646 IC50 = 15.7 nM T12541 CLNB61 134148636 IC50 = 59.2 nM T12541 CEPY30 134148697 IC50 = 208.5 nM T12541 CH9JD6 134148851 IC50 = 105.8 nM T12541 C2HA3X 134149528 IC50 = 8.6 nM T12541 C8ZPJ0 134150664 IC50 = 93.5 nM T12541 C4YG8O 134150788 IC50 = 39.4 nM T12541 CG8LE2 134151667 IC50 = 6.1 nM T12541 CZ9M1G 134152630 IC50 = 189.4 nM T12541 C0W2DJ 134152820 IC50 = 76.3 nM T12541 C8Q4BJ 134153296 IC50 = 41.5 nM T12541 C9R5ZB 134153378 IC50 = 13.4 nM T12541 CE2RO0 134155126 IC50 = 5.3 nM T12541 CT84VF 134155258 IC50 = 12.5 nM T12541 CYFU82 134155860 IC50 = 163.3 nM T12541 C8NYC5 134155918 IC50 = 9 nM T12541 C54FXD 134957362 IC50 > 10000 nM T12541 C8M3DS 135742054 IC50 = 5.7 nM T12541 CU29YK 135750268 IC50 = 1600 nM T12541 C12UDA 135947972 IC50 = 210 nM T12541 CN42ZS 135947973 IC50 = 2600 nM T12541 CF8AO3 135947974 IC50 = 470 nM T12541 CJN7E2 135947978 IC50 = 870 nM T12541 CFKH34 135947979 IC50 = 7400 nM T12541 CV3UE9 137333450 IC50 = 300.2 nM T12541 CS78JW 137639139 IC50 = 2800 nM T12541 C9O2PL 145958063 IC50 = 68 nM T12541 C9NS6T 145958690 IC50 = 114.5 nM T12541 CTJI01 145964752 IC50 = 11 nM T12541 CQZ3F7 145965198 IC50 = 8 nM T12541 CQH7A1 145966715 IC50 > 6000 nM T12541 C37OFS 145969385 IC50 > 10000 nM T12541 C2DL3V 145970081 IC50 = 3387 nM T12541 CQ1O4U 145973476 IC50 = 5743 nM T12541 C4OFQ8 145974197 IC50 = 173 nM T12541 CYEH74 145974272 IC50 = 1768 nM T12541 C2CTW7 145974410 IC50 = 42 nM T12541 CPM02H 145975616 IC50 = 2 nM T12541 CZQN94 145976919 IC50 = 380 nM T12541 CC2H5G 145977751 IC50 = 414 nM T12541 CWJ46S 145978007 IC50 = 7 nM T12541 C45VBD 155511230 IC50 = 5800 nM T12541 CV68FP 155518122 IC50 = 1360 nM T12541 C1N8GW 155518838 IC50 = 6980 nM T12541 C9LBF0 155519200 IC50 = 1540 nM T12541 C85WOD 155521426 IC50 = 9930 nM T12541 C2G6QJ 155526648 IC50 = 9520 nM T12541 CEB07F 155528709 IC50 = 140 nM T12541 C3Q9WN 155535344 IC50 = 90 nM T12541 CBR30A 155545077 IC50 = 4840 nM T12541 C36FGC 155545735 IC50 = 14160 nM T12541 C07GNA 155546020 IC50 = 600 nM T12541 C8ZC3B 155553069 IC50 = 3400 nM T12541 CBOJ62 155560887 IC50 = 2100 nM T12541 C5GL3E 155561063 IC50 = 5460 nM T12541 CKSD18 155561108 IC50 = 5390 nM T12541 CGK2P5 155565175 IC50 = 730 nM T12541 CLH4A2 155567806 IC50 = 1710 nM T12541 D03EHM 24905142 IC50 = 60 nM T12541 D06HVH 54613583 IC50 = 2500 nM T12541 D0H0HR 49836027 IC50 = 6680 nM T12541 D0H2CM 135565635 IC50 = 408 nM T12541 D0P5TI 58441401 IC50 > 1000 nM T12541 D0S5YV 6852167 IC50 = 19 nM T28893 D00JVR 2267 IC50 = 6309.57 nM T28893 D01AZG 5073 Ki > 1000 nM T28893 D01ZII 2726 Ki = 125.89 nM T28893 D02EYG 10096344 IC50 = 295 nM T28893 D04JEE 4946 EC50 > 5011.87 nM T28893 D06HLY 5910 EC50 = 17.5 nM T28893 D06MAJ 65906 Ki > 10000 nM T28893 D06XZR 27400 Ki = 2 nM T28893 D08CTT 21855 Ki = 263.03 nM T28893 D09VBC 2562 Ki = 76 nM T28893 D09ZOQ 11519069 Ki = 0.16 nM T28893 D0B4TN 2381 Ki = 2.36 nM T28893 D0BZ7W 443879 Ki = 1.4 nM T28893 D0D1AL 3559 Ki = 1600 nM T28893 D0E6YQ 1935 IC50 = 13000 nM T28893 D0G8NN 119570 Ki > 10000 nM T28893 D0H3HM 60795 Ki > 1000 nM T28893 D0H7KF 5002 Ki = 56 nM T28893 D0L4YD 154059 Ki = 51.29 nM T28893 D0M0AM 11693 IC50 = 0.1259 nM T28893 D0M6VK 71183 Ki = 0.0955 nM T28893 D0Q9HF 187 EC50 = 1.1 nM T28893 D0R1JV 60854 Ki = 5100 nM T28893 D0R7WU 1979 EC50 = 4466 nM T28893 D0RD5W 154417 Ki = 0.2692 nM T28893 D0RG3O 174174 Ki = 0.25 nM T28893 D0T0LM 4848 IC50 = 1.479 nM T28893 D0U5OE 3964 IC50 = 5500 nM T28893 D0U7BW 5831 Ki = 170 nM T28893 D0V4QS 135398745 Ki = 2.1 nM T28893 D0VP1V 11434515 Ki = 0.08 nM T28893 D0W8SJ 4199 Ki = 17000 nM T28893 D0Y5AM 444031 Ki = 5.5 nM T28893 D0Z1RV 135398737 Ki = 0.98 nM T28893 D02WFN 46207733 Ki = 8 nM T28893 D04YEW 25147683 IC50 = 0.9 nM T28893 D07EFM 2230 Ki = 14 nM T28893 D09JLI 3009355 Ki > 10000 nM T28893 D0I5XU 16065403 Ki = 0.115 nM T28893 D0K4HW 135409468 EC50 = 18 nM T28893 D0LI1C 44469321 IC50 > 10000 nM T28893 D02JNY 10030021 Ki = 316.23 nM T28893 D06ACX 6436265 Ki = 4.5 nM T28893 D06DZI 107780 Ki < 1000 nM T28893 D07IZF 9867750 Ki = 117 nM T28893 D08SOF 5405 IC50 = 2900 nM T28893 D08YVT 9894173 Ki = 653 nM T28893 D09FYQ 9577995 EC50 = 63.6 nM T28893 D0A2OW 107867 Ki = 179 nM T28893 D0A3OF 10026300 IC50 = 490 nM T28893 D0IE4H 131460 IC50 = 0.001 nM T28893 D0J8UV 9928284 EC50 = 41 nM T28893 D0PZ9R 45260374 EC50 = 1.1 nM T28893 D0R1VL 132712 Ki = 1071.52 nM T28893 D0S1VV 119053 IC50 = 3710 nM T28893 D0UX0T 9571002 EC50 = 21 nM T28893 D0VZ3D 129989 Ki = 28.84 nM T28893 C45PUM 2551 EC50 = 630.96 nM T28893 C4AWJ9 2684 Ki = 4897.79 nM T28893 C0H8GR 3191 IC50 = 1100 nM T28893 CFS16G 3450 Ki = 8511.38 nM T28893 CKD46H 4022 Ki = 1949.84 nM T28893 C7VMZ3 4108 Ki = 49.8 nM T28893 C2AF8D 6060 EC50 = 770 nM T28893 C5H9CN 9287 Ki > 10000 nM T28893 CV42HF 16817 EC50 = 5300 nM T28893 CVJ8F2 17931 EC50 > 10000 nM T28893 C89UZB 18493 Ki = 1.59 nM T28893 CL9I7S 19716 IC50 = 2450 nM T28893 CXFM39 39762 EC50 = 777 nM T28893 CRCD50 60809 IC50 = 0.008 nM T28893 C8E9XD 66007 IC50 = 1.3 nM T28893 C97NOS 68634 EC50 = 400 nM T28893 C3WKC6 68835 IC50 > 100000 nM T28893 C3S8RF 71792 EC50 = 820 nM T28893 C6ZQ4D 72064 Ki = 271 nM T28893 CA3W0P 100826 IC50 > 100000 nM T28893 CQA93V 118500 Ki = 740 nM T28893 C27RUO 129486 Ki = 0.088 nM T28893 CG56JL 129993 Ki = 6300 nM T28893 C2WO0V 163938 IC50 = 400 nM T28893 CVWA68 197841 Ki = 5.78 nM T28893 CZ0UI5 208598 Ki = 10000 nM T28893 CHLK79 214124 Ki = 4 nM T28893 C71KVJ 275176 Ki = 176 nM T28893 CD65GI 315401 Ki = 1.29 nM T28893 C1C2JH 372625 Ki = 3.981 nM T28893 C6OQ8S 410345 Ki = 7.75 nM T28893 CJ1QN5 425249 Ki = 971 nM T28893 C4J8NF 483747 Ki = 575 nM T28893 CFJ63U 511332 Ki = 350 nM T28893 CX75UZ 598754 Ki > 19952.62 nM T28893 CC56KR 639794 Ki = 12022.64 nM T28893 C91GCI 657308 Ki = 0.433 nM T28893 CEGR96 657346 Ki = 10964.78 nM T28893 C04XRI 657347 Ki = 10964.78 nM T28893 CYO7F3 688566 IC50 = 0.36 nM T28893 C4HCK5 729510 IC50 > 30000 nM T28893 CZN6S9 743974 EC50 > 15848.93 nM T28893 CR0E8B 826706 EC50 = 180 nM T28893 C08WCU 851833 Ki > 19952.62 nM T28893 CO59NV 939077 IC50 = 0.31 nM T28893 CUD48J 952858 IC50 = 3200 nM T28893 CZ6Q4Y 1090198 IC50 = 3200 nM T28893 C4O6ZA 1090202 IC50 = 960 nM T28893 CWFV17 1392038 IC50 = 2100 nM T28893 CH5WR4 1421986 IC50 = 2900 nM T28893 CPWD47 1956898 IC50 = 180 nM T28893 CS8N5X 2736067 Ki = 7943.28 nM T28893 C9NDW0 2802905 EC50 > 10000 nM T28893 CUF0Z9 3009352 Ki = 3900 nM T28893 CMK58I 3009353 Ki = 6075 nM T28893 CPN54Q 3009354 Ki > 3900 nM T28893 C6ZYX5 3009356 Ki = 1894 nM T28893 C5X0LK 3009357 Ki > 3700 nM T28893 C5NL4Z 3081966 EC50 = 317 nM T28893 C7ET2M 3156646 IC50 = 820 nM T28893 CMCH82 3242997 IC50 > 10000 nM T28893 CJ6D8N 3342390 Ki < 1000 nM T28893 CI7DF6 3675988 Ki = 177827.94 nM T28893 CX3S8T 4715419 Ki = 38018.94 nM T28893 C12BJA 4995951 Ki = 1318.26 nM T28893 CS71UA 5189681 IC50 > 30000 nM T28893 CR5LG3 5310989 IC50 = 5616.8 nM T28893 CQ45UT 5377745 EC50 = 3678 nM T28893 C83CEP 5378491 EC50 = 4479 nM T28893 CIO5H6 5379120 EC50 = 962 nM T28893 C1P3QG 5487543 IC50 = 7680 nM T28893 C07PJQ 6603753 Ki = 10964.78 nM T28893 C3A1FO 6604789 Ki = 10000 nM T28893 CFN7L4 6604866 Ki = 190.55 nM T28893 C2IP0Y 7022778 Ki = 63095.73 nM T28893 CVSC58 7047822 Ki = 46773.51 nM T28893 C32TSZ 7141654 Ki = 154881.66 nM T28893 C7NJZ2 7141656 Ki = 14454.4 nM T28893 C8Z3VW 9154093 EC50 = 473 nM T28893 CYH05F 9794266 Ki = 2000 nM T28893 CEDB68 9798900 IC50 = 3 nM T28893 CL94XF 9799291 Ki = 6.6 nM T28893 C8XGV3 9804849 IC50 = 1300 nM T28893 C7MBO3 9809330 Ki = 0.1 nM T28893 CX3U7N 9813501 Ki = 1200 nM T28893 CJM0W8 9816863 Ki = 6100 nM T28893 CMC3O6 9821459 Ki = 19 nM T28893 C6NJO3 9827782 Ki = 6.486 nM T28893 CLX9T1 9838314 EC50 > 10000 nM T28893 CH74OS 9846311 Ki = 1.5 nM T28893 CB31LS 9855978 Ki = 1900 nM T28893 CTUM52 9856417 Ki = 1100 nM T28893 C3YI2L 9857572 IC50 = 1.1 nM T28893 CGO07X 9859365 Ki = 9.6 nM T28893 CSTG23 9866745 IC50 = 84 nM T28893 C1N0KW 9867847 Ki = 2.8 nM T28893 CQ4LC2 9872676 Ki = 4120 nM T28893 CL0VY5 9874177 Ki = 1.9 nM T28893 CYSB08 9878065 Ki = 2600 nM T28893 C19JZH 9883040 Ki = 124 nM T28893 CJ5K1D 9889312 Ki = 83 nM T28893 CR5PO3 9903030 IC50 = 39.7 nM T28893 C0YG4J 9904307 EC50 = 164.8 nM T28893 C2U5LK 9905467 IC50 = 14.5 nM T28893 CF49JB 9905609 Ki > 1400 nM T28893 CCT20X 9905731 Ki = 58 nM T28893 C0ZQ3O 9905964 Ki = 112 nM T28893 CYWQ50 9906447 Ki = 3266 nM T28893 CDB9E1 9909907 Ki = 50.12 nM T28893 CL5HA4 9910802 Ki = 5.3 nM T28893 CXAV92 9911615 Ki = 3311.31 nM T28893 C9OK6J 9912392 Ki = 1.2 nM T28893 CXAY37 9913341 Ki = 50.12 nM T28893 C6EK8M 9916275 Ki > 1000000 nM T28893 CQ3L1X 9921302 Ki = 2500 nM T28893 CJ46NU 9921303 Ki = 150 nM T28893 CBE1Y9 9921863 Ki = 3800 nM T28893 C9W7OU 9926604 Ki = 7 nM T28893 CG4PD5 9927975 EC50 = 0.2 nM T28893 C3L5GV 9928017 IC50 = 0.4 nM T28893 CRV17M 9931930 Ki = 2041.74 nM T28893 C50NSR 9936450 Ki = 0.84 nM T28893 CA2HR0 9937709 Ki = 1.6 nM T28893 C5E7KC 9943680 Ki = 6500 nM T28893 C65PMK 9944783 IC50 = 0.8 nM T28893 C36NIB 9946010 IC50 = 0.4 nM T28893 CY4L1D 9946632 IC50 = 8.3 nM T28893 CUCT38 9948957 Ki = 910 nM T28893 CMO0X9 9949717 EC50 = 210 nM T28893 C7TD1E 9953227 Ki = 4.4 nM T28893 CWSE34 9954899 IC50 > 1000 nM T28893 C8BD2S 9956104 Ki = 4.9 nM T28893 C58KXV 9958728 Ki = 0.23 nM T28893 C1X7FR 9960272 Ki = 1.5 nM T28893 C4I7UJ 9964754 Ki = 870 nM T28893 CFG21X 9966959 IC50 = 0.8 nM T28893 CH23EP 9967590 IC50 = 0.4 nM T28893 CYNT43 9968046 Ki = 1737.8 nM T28893 CCM72P 9974222 IC50 = 9.6 nM T28893 CT26UJ 9974229 Ki = 222 nM T28893 CMY73F 9978490 IC50 = 170 nM T28893 CF41ZD 9980157 IC50 = 401 nM T28893 C6QZ8W 9984928 Ki = 31.7 nM T28893 C3G0VC 9985181 Ki = 59.4 nM T28893 C9XS0E 9990434 EC50 = 4700 nM T28893 CD9A5M 9991939 Ki = 81 nM T28893 C8F4XT 9991979 Ki = 170 nM T28893 CYK1U4 9996901 IC50 = 34.8 nM T28893 C9FR0C 9998508 Ki = 891.25 nM T28893 C17BCF 10003476 IC50 = 1190 nM T28893 CN8XI3 10006926 IC50 = 1174 nM T28893 CK19GL 10007637 IC50 = 1 nM T28893 CV0KA3 10019339 EC50 = 4.9 nM T28893 C6V3NE 10020614 Ki = 135 nM T28893 CQZ0K4 10027177 EC50 = 334 nM T28893 C7I6DA 10035281 Ki = 2300 nM T28893 CO69GW 10035533 IC50 = 216 nM T28893 CBJ63D 10043954 Ki = 1479.11 nM T28893 CX27EK 10049758 IC50 = 460 nM T28893 C56FEU 10053613 IC50 = 4.4 nM T28893 C9Z3TI 10058347 IC50 = 216 nM T28893 C2WJS1 10058649 Ki = 360 nM T28893 CORA81 10058744 IC50 = 2590 nM T28893 CV6A5I 10061123 Ki = 820 nM T28893 C9OQ2S 10066369 Ki = 741.31 nM T28893 CI6SD7 10066972 Ki = 1258.93 nM T28893 C1GUM0 10080742 IC50 = 4050 nM T28893 C6Z5CY 10081053 IC50 = 3840 nM T28893 CCO72H 10082470 IC50 = 1800 nM T28893 CQ3O0X 10085070 IC50 = 1090 nM T28893 C8NQ3I 10092649 EC50 = 6.5 nM T28893 C42OHV 10093490 EC50 = 880 nM T28893 C4IZ5H 10101246 Ki = 0.01288 nM T28893 CT4XE6 10103909 Ki = 2200 nM T28893 CHUE04 10104527 Ki = 9200 nM T28893 COR41M 10105880 Ki = 1800 nM T28893 CG0O9Z 10109893 EC50 = 794.33 nM T28893 CUT05R 10114698 Ki = 20417.38 nM T28893 C9XDU8 10119938 IC50 = 1.6 nM T28893 C20GMN 10132599 IC50 = 1 nM T28893 CFH60N 10133281 IC50 = 2.4 nM T28893 C0V1PA 10138000 Ki = 398.11 nM T28893 C90FZG 10139614 Ki = 3090.3 nM T28893 C0PO3J 10142923 Ki = 25.12 nM T28893 CPF96U 10143717 IC50 = 0.4 nM T28893 CC8YJ1 10143857 IC50 = 2 nM T28893 C7LP4V 10143953 IC50 = 0.81 nM T28893 CYU79M 10143955 Ki = 0.09 nM T28893 CG78WP 10160073 Ki = 13180 nM T28893 CZ8E9X 10160219 Ki = 870.96 nM T28893 CVI4O6 10164136 IC50 = 1.4 nM T28893 CXCT70 10165876 IC50 = 0.4 nM T28893 CQA5E4 10179727 Ki = 79.43 nM T28893 C4TR5Q 10180872 Ki = 6 nM T28893 C1N4VJ 10182489 Ki = 199.53 nM T28893 C1B8RO 10187215 IC50 = 1.4 nM T28893 C0JS1M 10198147 IC50 ~ 10000 nM T28893 COR14Y 10203251 Ki = 1318.26 nM T28893 CB69ND 10204457 Ki = 71.8 nM T28893 CUW93D 10208896 IC50 = 1.5 nM T28893 C57WMS 10208971 IC50 = 1.7 nM T28893 C0G2IA 10220374 IC50 = 52.48 nM T28893 C2H1WR 10220392 EC50 = 3300 nM T28893 CJ5V2S 10225340 Ki = 31.09 nM T28893 C04QCB 10225881 Ki = 870.96 nM T28893 C6A5KD 10226456 Ki = 3.981 nM T28893 C8XY5N 10229166 IC50 = 2 nM T28893 CO64WJ 10236758 EC50 = 34.67 nM T28893 CRQ8D4 10240891 IC50 = 26900 nM T28893 CE69PK 10242813 Ki = 100 nM T28893 CQB1O6 10243426 Ki = 37 nM T28893 CEYJ57 10244370 Ki = 1200 nM T28893 C49MUR 10246307 IC50 = 0.4 nM T28893 C3W2YB 10248541 IC50 = 1410 nM T28893 C3QGA5 10251795 EC50 = 260 nM T28893 C2LK8V 10256272 IC50 = 114 nM T28893 CW90FO 10261985 EC50 = 140 nM T28893 CLS61Z 10262405 IC50 = 9640 nM T28893 C1FCP7 10262466 Ki = 905 nM T28893 CC6RP7 10267601 IC50 = 18.1 nM T28893 CY3E5J 10274019 Ki = 0.53 nM T28893 C7CYM8 10275847 Ki = 16.4 nM T28893 CG6I4F 10299489 Ki = 23 nM T28893 C7WMZ6 10300660 IC50 = 2.5 nM T28893 CB83CP 10313301 Ki = 26000 nM T28893 CD1C0H 10315426 Ki = 3235.94 nM T28893 CF05IP 10324012 Ki = 68.08 nM T28893 CWP67J 10330721 Ki = 11600 nM T28893 CLW9R8 10330893 Ki = 220 nM T28893 CYIS62 10333583 IC50 = 1120 nM T28893 C3E5CB 10337773 Ki = 25118.86 nM T28893 C9YR5B 10339062 Ki = 520 nM T28893 C6S7GK 10354348 IC50 > 100000 nM T28893 C5M9WO 10354430 Ki = 810 nM T28893 C5UTA9 10356006 IC50 = 3340 nM T28893 CY3R2L 10356836 IC50 = 5100 nM T28893 CP0LR5 10357756 Ki > 10000 nM T28893 C7BZ1R 10358345 IC50 = 35 nM T28893 CBSA40 10360219 Ki = 426.58 nM T28893 CLM8P2 10365639 Ki = 6.98 nM T28893 CR0QC5 10367502 IC50 = 430 nM T28893 C9LWG3 10369004 IC50 = 670 nM T28893 CY9G0R 10375322 EC50 = 5900 nM T28893 CUD07Z 10376012 EC50 = 5050 nM T28893 CXN2K4 10376182 IC50 = 7890 nM T28893 C72EML 10392704 IC50 = 53.8 nM T28893 C85QEA 10397133 EC50 = 890 nM T28893 C5TX2E 10397356 EC50 = 1900 nM T28893 CUBA69 10398843 Ki = 57 nM T28893 CQW10P 10399393 EC50 = 5100 nM T28893 C54MOT 10403330 EC50 = 135.8 nM T28893 C30DKF 10405613 Ki = 82.4 nM T28893 CALE73 10419574 EC50 = 27000 nM T28893 CID42C 10420458 IC50 = 1580 nM T28893 C0IPX1 10421689 Ki = 410 nM T28893 CL7D2U 10421982 Ki = 270 nM T28893 C07QHE 10429011 Ki = 360 nM T28893 C5BEJ0 10442081 EC50 = 460 nM T28893 CIRS06 10442337 EC50 = 95 nM T28893 CZU94X 10444753 EC50 = 31 nM T28893 CS63AC 10447114 Ki > 10000 nM T28893 CAW4U0 10451242 EC50 = 7.6 nM T28893 CA3CY4 10451634 Ki = 75 nM T28893 C4C7UG 10457079 Ki = 0.007943 nM T28893 CI8R9A 10465050 Ki = 1200 nM T28893 CC9AV4 10465280 EC50 = 170 nM T28893 C6B5DJ 10465524 IC50 = 9440 nM T28893 CK9ZH7 10466231 Ki = 34 nM T28893 CVK48E 10467755 Ki = 1100 nM T28893 C53SCK 10468535 Ki = 50 nM T28893 CA14ZS 10468764 IC50 = 36300 nM T28893 CE6JH3 10473919 Ki = 1058 nM T28893 C26BIM 10475156 Ki = 3800 nM T28893 CEF2O6 10478367 Ki > 10000 nM T28893 C1GT3O 10487582 IC50 = 1180 nM T28893 C8COH6 10499832 IC50 = 670 nM T28893 C18ZYN 10500741 Ki = 2.6 nM T28893 CU0B8N 10501523 Ki = 1200 nM T28893 CO62HL 10503358 Ki = 0.88 nM T28893 CS1P4M 10511551 IC50 = 1500 nM T28893 CKP8N1 10515352 IC50 = 4030 nM T28893 CP9M5J 10516408 IC50 = 291.2 nM T28893 C37PDA 10518821 IC50 = 19027.3 nM T28893 C6T1JW 10521205 IC50 = 105.2 nM T28893 C4WZ3R 10522202 IC50 = 610.6 nM T28893 C5MB2F 10522336 IC50 = 30.4 nM T28893 C3EZ5Y 10525412 Ki = 3.5 nM T28893 C0K9HN 10538337 IC50 = 33117.6 nM T28893 CD9RI5 10539130 IC50 = 5460 nM T28893 C3Y6JB 10546275 IC50 = 11.5 nM T28893 CI3GQ6 10547222 IC50 = 484.2 nM T28893 C6XKZ9 10549581 IC50 = 4024.4 nM T28893 CSC81Z 10551354 Ki = 2.5 nM T28893 CUJ3W9 10563152 IC50 = 9850 nM T28893 CFD40Z 10567192 IC50 = 16.9 nM T28893 C4AL8Q 10569816 IC50 = 93.5 nM T28893 CHI03M 10572657 Ki = 470 nM T28893 C0Z5PY 10572658 Ki = 660 nM T28893 CV62YH 10573458 Ki = 36 nM T28893 CB37SH 10573693 IC50 = 2829.7 nM T28893 CR2GX4 10574041 Ki = 72 nM T28893 C71VMD 10591874 IC50 = 65.4 nM T28893 C94VUE 10592484 IC50 = 161.4 nM T28893 C51LBK 10593954 IC50 = 59.2 nM T28893 CH2QU8 10594386 IC50 = 963.2 nM T28893 CY54RA 10595006 Ki = 170 nM T28893 C6VGM0 10597259 Ki = 75 nM T28893 CVY63G 10598540 Ki = 70 nM T28893 CZRJ60 10610375 IC50 = 2308 nM T28893 C5HKT1 10610448 IC50 = 1620 nM T28893 CX01SE 10611310 IC50 = 888.1 nM T28893 CO3H7D 10614695 IC50 = 1819.5 nM T28893 C3BK2J 10619926 Ki = 140 nM T28893 C34LMA 10621363 Ki = 1.4 nM T28893 CSGO98 10622033 Ki = 22 nM T28893 C92HRJ 10622718 Ki = 140 nM T28893 CLJ29W 10623721 Ki = 340 nM T28893 CJL4R1 10636001 IC50 = 278 nM T28893 C09XHV 10638050 IC50 = 84.8 nM T28893 C5VWL8 10641009 IC50 = 38.7 nM T28893 C2ZTE6 10646906 Ki = 3.5 nM T28893 CDAG26 10646948 Ki = 1.2 nM T28893 CZ7M1D 10647553 Ki = 17 nM T28893 CX49UY 10647703 Ki = 2.5 nM T28893 CJG5D4 10657039 EC50 = 6202 nM T28893 CONH15 10663572 IC50 = 13.4 nM T28893 C6WQ2Z 10664532 IC50 = 233.6 nM T28893 C8CF4H 10666533 IC50 = 159 nM T28893 C56EGM 10670917 Ki = 3.2 nM T28893 C1DSK6 10670961 Ki = 14 nM T28893 CUYW18 10671167 Ki = 170 nM T28893 C0AV8X 10678449 IC50 = 10000 nM T28893 C32KQX 10684720 IC50 = 67.9 nM T28893 CZQY38 10686494 IC50 = 37.15 nM T28893 C32EGP 10686988 IC50 = 61.4 nM T28893 C9O6LN 10688349 IC50 = 3285.2 nM T28893 C6PDH5 10693031 Ki = 2.1 nM T28893 CW91HU 10707175 IC50 = 16600 nM T28893 C62MCG 10716120 Ki = 61 nM T28893 CS3W1G 10718110 Ki = 26 nM T28893 CEB3A5 10726038 IC50 = 1650 nM T28893 C5OF4K 10739662 Ki = 200 nM T28893 CC21XD 10755732 IC50 = 76.8 nM T28893 CHL29Z 10755733 IC50 = 120.5 nM T28893 C4JXA3 10757736 IC50 = 1141.1 nM T28893 C15WSV 10759971 Ki = 65.9 nM T28893 CPQ7Z3 10760249 IC50 = 8.8 nM T28893 C5P3DQ 10761219 IC50 = 743.1 nM T28893 CTNG89 10777343 IC50 = 14100 nM T28893 CX4LT3 10777692 IC50 = 2220.1 nM T28893 CC7TL1 10778462 IC50 = 10600 nM T28893 CU5SO1 10778750 IC50 = 4010 nM T28893 CA4QI2 10782321 IC50 = 888.6 nM T28893 C4N9IT 10782462 IC50 = 54.2 nM T28893 C6FC0M 10784004 IC50 = 122 nM T28893 CV8TE0 10785471 IC50 = 106.1 nM T28893 CW5TJ6 10797864 IC50 = 99 nM T28893 C5FVW2 10800287 EC50 = 4867 nM T28893 C9SEA6 10806268 IC50 = 78 nM T28893 CGR64V 10808719 IC50 = 69.4 nM T28893 C3QK4R 10810094 Ki = 4300 nM T28893 CR4XK8 10812455 Ki = 2.4 nM T28893 CX9B7I 10826990 IC50 = 15100 nM T28893 CK1D3J 10827157 IC50 = 128 nM T28893 C4I3MN 10828627 IC50 = 37 nM T28893 CR1X5L 10829928 IC50 = 1087.7 nM T28893 C0GS8Z 10830843 Ki = 310 nM T28893 C2M0QO 10834711 Ki = 9 nM T28893 C27NPT 10835518 Ki = 200 nM T28893 C2S6DG 10836338 Ki = 15 nM T28893 CB7E2O 10846833 IC50 = 20500 nM T28893 CFQ74S 10848032 IC50 = 4840 nM T28893 CH9WK6 10851853 IC50 = 63.7 nM T28893 CX6AP3 10852843 IC50 = 913.1 nM T28893 C5PRT6 10854879 IC50 = 77.3 nM T28893 C8HI5L 10854880 IC50 = 22 nM T28893 CZ85AJ 10862395 Ki = 2187.76 nM T28893 CHE9P4 10865439 Ki = 108 nM T28893 CCM3L9 10870954 Ki = 16218.1 nM T28893 C2YNC5 10871551 Ki = 223.87 nM T28893 CFAD04 10874119 Ki = 1174.9 nM T28893 CTV95B 10880435 Ki = 1584.89 nM T28893 CFP75Y 10907744 Ki = 0.61 nM T28893 C4A8QE 10916286 Ki > 4365.16 nM T28893 CQLR32 10919522 Ki = 14 nM T28893 CC12TE 10925451 Ki = 346.74 nM T28893 C2ZX9Q 10929712 Ki = 0.93 nM T28893 CU09AV 10937901 IC50 = 630 nM T28893 CSLT97 10949380 IC50 = 556 nM T28893 C5LVY0 10949838 Ki = 1513.56 nM T28893 CE05FM 10951142 Ki = 363.08 nM T28893 C1WF5L 10952349 Ki = 0.32 nM T28893 CA6X3W 10952416 Ki = 0.57 nM T28893 C3K6JV 10957754 Ki = 891.25 nM T28893 CGBA73 10962438 Ki = 20 nM T28893 CN4QT5 10963509 Ki = 19.8 nM T28893 C4WV8L 10969390 Ki = 602.56 nM T28893 CTYZ13 10969696 Ki = 4365.16 nM T28893 C41PXY 10982070 Ki = 1174.9 nM T28893 C9E2MP 10984804 Ki > 2500 nM T28893 CZXG56 10984923 Ki = 5 nM T28893 C2W3GM 11000399 Ki = 4265.8 nM T28893 C6NH9T 11001809 Ki = 3548.13 nM T28893 CQ8D4K 11004046 Ki = 1995.26 nM T28893 CK3RT9 11006286 Ki = 14 nM T28893 C6BG1N 11006792 Ki = 150 nM T28893 CU4Z0J 11011332 Ki = 3715.35 nM T28893 CZK86F 11011757 Ki = 158.49 nM T28893 CVA6U9 11012653 Ki = 870.96 nM T28893 CPM1Z7 11012712 Ki = 1548.82 nM T28893 CW23BJ 11013666 Ki = 43.65 nM T28893 C6TF5I 11015312 Ki = 1318.26 nM T28893 C7Y1DO 11024241 Ki = 870.96 nM T28893 C3L9ON 11034265 Ki = 331.13 nM T28893 CHDT49 11039424 Ki = 120 nM T28893 CP9OJ6 11045444 Ki = 245.47 nM T28893 C4ZUH9 11048067 Ki = 1318.26 nM T28893 CQ8O3Y 11057942 Ki > 21877.62 nM T28893 CIG31V 11061341 Ki = 150 nM T28893 CT3XN5 11071537 EC50 = 398.11 nM T28893 CO3C6Q 11072401 Ki = 0.69 nM T28893 C5VQ6H 11079969 Ki = 1318.26 nM T28893 CWS56C 11092603 Ki = 199.53 nM T28893 C02MPO 11099206 Ki = 1047.13 nM T28893 CSNA03 11101362 Ki = 5128.61 nM T28893 CF81CB 11110049 Ki = 53703.18 nM T28893 C7ROJ1 11112362 Ki = 2511.89 nM T28893 C9CY0M 11120347 Ki = 562.34 nM T28893 CD20CQ 11120503 EC50 = 67.3 nM T28893 C8ITB9 11124824 Ki = 7.6 nM T28893 C2C4AN 11131099 Ki = 3715.35 nM T28893 CB37ZA 11135606 Ki = 0.19 nM T28893 C1T9WI 11143997 Ki = 1778.28 nM T28893 CX69QO 11223597 Ki = 0.38 nM T28893 C92CYH 11265950 Ki = 19 nM T28893 C4S2VF 11277147 Ki > 1000 nM T28893 CSH2N3 11294846 IC50 > 5000 nM T28893 CI1EN4 11306851 IC50 = 3.1 nM T28893 CT6MF7 11316670 IC50 = 954 nM T28893 CBR60Z 11318734 IC50 = 158.49 nM T28893 CE3O6K 11386357 IC50 = 5607 nM T28893 CR9EB8 11396245 IC50 = 2804 nM T28893 C85LYP 11430418 IC50 > 1000 nM T28893 C9FNM4 11431811 Ki = 0.013 nM T28893 CGD57K 11431873 Ki = 0.12 nM T28893 C9NUV4 11442477 IC50 = 1.6 nM T28893 CIN42A 11489418 IC50 = 0.41 nM T28893 C1O9XD 11493620 Ki > 10000 nM T28893 C69AMJ 11500781 Ki > 10000 nM T28893 CTVZ02 11503335 IC50 = 2.7 nM T28893 CLPO39 11508317 Ki = 5.8 nM T28893 CBZ5E8 11508710 IC50 = 45.1 nM T28893 CSP02B 11510357 IC50 = 12.2 nM T28893 CDQ18N 11515125 IC50 > 10000 nM T28893 CP9RB7 11515387 Ki > 10000 nM T28893 CGCF61 11515738 Ki < 100000 nM T28893 C7OKD1 11518067 IC50 = 2.4 nM T28893 CY63VP 11523050 Ki = 93325.43 nM T28893 C0BC6Y 11530223 Ki > 10000 nM T28893 C07AJD 11530306 Ki < 100000 nM T28893 C89JTB 11532924 Ki = 260 nM T28893 CR17KT 11535021 EC50 = 36307.81 nM T28893 CQ08DH 11539632 IC50 = 1.7 nM T28893 CWUP85 11542982 Ki < 100000 nM T28893 C0ZF8J 11544156 Ki = 2 nM T28893 C6B2XK 11547052 IC50 = 5.8 nM T28893 C34JAV 11551351 Ki = 990 nM T28893 CNZJ38 11552174 IC50 = 19.1 nM T28893 CP9UJ1 11569907 IC50 = 0.44 nM T28893 CP04FM 11569925 IC50 = 15.1 nM T28893 CXP2M0 11580426 Ki = 1400 nM T28893 CW7G3X 11580427 Ki = 5.3 nM T28893 CYW90N 11583261 IC50 = 2.6 nM T28893 C6D1MA 11584660 IC50 = 1584.89 nM T28893 CEHP14 11586481 Ki < 100000 nM T28893 CP3Y7J 11588240 Ki < 100000 nM T28893 C43RFK 11600183 EC50 = 8912.51 nM T28893 CP3G5L 11602980 IC50 = 13.8 nM T28893 C15DMA 11617374 IC50 = 73.8 nM T28893 CE07UT 11619197 IC50 = 4.5 nM T28893 CQ5PI4 11622544 Ki < 100000 nM T28893 C79OMR 11623756 IC50 = 4700 nM T28893 CSB9O5 11623845 Ki = 2072000 nM T28893 CK4GS9 11626846 IC50 = 3.8 nM T28893 CZ4QC1 11635866 Ki > 10000 nM T28893 C23XSL 11638166 Ki = 5.6 nM T28893 C4FK7Z 11651028 Ki = 29.4 nM T28893 C3RV2P 11651045 Ki = 189 nM T28893 CF2ZC0 11651360 Ki < 100000 nM T28893 CHKN81 11653111 Ki < 100000 nM T28893 C1HDM5 11653679 Ki = 871.6 nM T28893 CH3N1I 11659592 Ki = 28000 nM T28893 C27XOS 11660220 Ki < 100000 nM T28893 C0N4BQ 11672895 Ki < 100000 nM T28893 C0ZK8U 11678377 IC50 = 4.9 nM T28893 CN4Z5C 11679149 IC50 > 10000 nM T28893 C7JVX2 11681378 Ki > 10000 nM T28893 CY36RI 11688223 Ki > 10000 nM T28893 CI5B1R 11690967 IC50 = 2.1 nM T28893 CQD96L 11691949 Ki = 0.64 nM T28893 CW8CE2 11694118 Ki < 100000 nM T28893 CF8MO2 11694119 Ki < 100000 nM T28893 CEQ6W7 11694810 Ki > 1000 nM T28893 C7Z0SX 11695591 Ki > 10000 nM T28893 CMT6F0 11695697 IC50 = 13.4 nM T28893 CP3G0Q 11695811 Ki > 10000 nM T28893 C3TN1P 11700268 Ki > 10000 nM T28893 CBDC74 11702114 Ki > 10000 nM T28893 CQ5P2F 11702115 Ki > 10000 nM T28893 CXFK83 11702578 Ki > 10000 nM T28893 CY31MF 11712407 IC50 = 15.8 nM T28893 C9BF1S 11715398 Ki < 100000 nM T28893 C24CMZ 11723664 Ki = 50 nM T28893 C0E9SG 11725107 EC50 = 20.2 nM T28893 C0O2QC 11725334 IC50 = 0.9 nM T28893 CEY7J3 11729182 Ki = 21877.62 nM T28893 CV7WM2 11734822 Ki = 17 nM T28893 CPG15O 11743399 IC50 > 1000 nM T28893 C4QVR6 11748799 Ki = 52.48 nM T28893 CQLP36 11759058 Ki = 48977.88 nM T28893 CW3GA7 11759212 Ki = 151.36 nM T28893 CBM05D 11759379 Ki = 1905.46 nM T28893 CFZ4L5 11767229 Ki = 110 nM T28893 C39HRB 11793999 IC50 = 316.7 nM T28893 CM16WE 11794901 Ki = 26 nM T28893 CT8P7Q 11796409 Ki = 57 nM T28893 C91DQM 11796509 Ki = 8.5 nM T28893 CHEA80 11798126 Ki = 4.4 nM T28893 CT4F2C 11808040 Ki = 34.67 nM T28893 CXQ10I 11808946 Ki = 239.88 nM T28893 C6EXD3 11808947 Ki = 229.09 nM T28893 C30WRH 11809446 Ki = 5370.32 nM T28893 CV43DH 11813912 Ki = 0.87 nM T28893 CF1S7Q 11819427 IC50 = 2610 nM T28893 C3MQW7 11819545 Ki = 1500 nM T28893 CQW16Z 11819782 Ki = 52480.75 nM T28893 C0BPK3 11819882 Ki = 290 nM T28893 C2KW3U 11819883 Ki = 710 nM T28893 CJIA51 11828362 Ki = 36 nM T28893 CR9FJ2 11833737 Ki = 1621.81 nM T28893 CZ3AX9 11834199 Ki = 446.68 nM T28893 C8JQL7 11957735 IC50 > 10000 nM T28893 CL91TM 11968014 IC50 = 1.514 nM T28893 CZAV59 12016985 EC50 > 10000 nM T28893 C5P3XD 12586122 Ki = 26000 nM T28893 CPA39N 12612376 EC50 = 870 nM T28893 CI60QE 12947027 EC50 = 516 nM T28893 CNVA43 13218688 Ki = 550 nM T28893 CR10FQ 13567080 Ki = 1.096 nM T28893 CW1PU9 14042939 EC50 > 10000 nM T28893 C19BYU 14479864 IC50 < 1 nM T28893 CS54WY 14537188 Ki = 0.881 nM T28893 CA87RQ 14660293 IC50 = 100000 nM T28893 CMFD17 14685518 Ki = 30000 nM T28893 CU36CN 14685523 Ki = 540 nM T28893 CR2O6Z 14851833 EC50 = 2154 nM T28893 CMO81H 14925759 EC50 = 645.65 nM T28893 CKWQ92 14936861 IC50 = 537 nM T28893 C6QNU8 15033741 IC50 = 3 nM T28893 CVNK57 15065550 Ki = 120.23 nM T28893 CZS96E 15105207 Ki > 10000 nM T28893 C38UHI 15105209 Ki = 1697 nM T28893 C49DYR 15105211 Ki = 843 nM T28893 CZ16XJ 15157137 Ki = 1.9 nM T28893 C5VC9Z 15157138 Ki = 2.9 nM T28893 C7VT5X 15157139 Ki = 40.7 nM T28893 CD3MI7 15157140 Ki = 111 nM T28893 CY80DC 15157141 Ki = 298 nM T28893 C4MZ1N 15180164 IC50 = 224 nM T28893 CAF40B 15181802 IC50 = 46 nM T28893 CSA5Y2 15196231 Ki > 15000 nM T28893 CO4EB0 15196232 Ki = 14900 nM T28893 COIG73 15196233 Ki = 7400 nM T28893 C80ICP 15196234 Ki = 300 nM T28893 CIV27H 15196235 Ki = 2200 nM T28893 CXZB18 15196236 Ki = 59 nM T28893 CEH60Q 15196354 Ki = 1100 nM T28893 CN1RW5 15392110 Ki = 1.3 nM T28893 CLNS53 15485015 IC50 = 809 nM T28893 C5PU2X 15521599 IC50 = 39 nM T28893 CO19UA 15595033 Ki = 988 nM T28893 C9C6WP 15629515 Ki > 50000 nM T28893 C4PYE0 15681299 IC50 = 1110 nM T28893 C48IJQ 15681300 IC50 = 3690 nM T28893 C0T6NK 15681301 IC50 = 14450 nM T28893 CG0RN6 15681303 IC50 = 42400 nM T28893 CEW1M8 15749863 Ki = 9300 nM T28893 CJ5Z9T 15749864 Ki = 19000 nM T28893 CK4JY7 15860348 EC50 = 102 nM T28893 CIW40C 15888010 Ki = 3 nM T28893 CJKM40 15888011 Ki = 0.98 nM T28893 CT64BE 15945874 IC50 = 1995.26 nM T28893 CUB5X2 16038385 EC50 = 63.1 nM T28893 CZ47FJ 16071018 EC50 = 5.012 nM T28893 C3T0UX 16085999 Ki = 300 nM T28893 CWI32N 16086000 Ki = 270 nM T28893 C71HBL 16086001 Ki = 65 nM T28893 C7EM1G 16086003 Ki = 1800 nM T28893 CFU72Z 16086004 Ki > 2600 nM T28893 CTOM27 16086005 Ki = 260 nM T28893 C7WF9Y 16086059 Ki = 170 nM T28893 C05YVJ 16086060 Ki = 300 nM T28893 CMQ8U3 16086061 Ki = 580 nM T28893 CEI8G1 16086062 Ki = 220 nM T28893 CGB89M 16086063 Ki = 71 nM T28893 CUS73E 16086064 Ki = 210 nM T28893 CHJ07L 16086065 Ki = 2000 nM T28893 CEV68D 16086066 Ki = 93 nM T28893 CIX9M7 16086067 Ki = 460 nM T28893 CEVD42 16091071 Ki = 2540 nM T28893 C1XZ7V 16094783 Ki = 794.33 nM T28893 CO16DS 16094788 EC50 = 251.19 nM T28893 CYN71L 16094791 Ki = 316.23 nM T28893 C2HK7W 16094793 Ki = 63.1 nM T28893 C9R0JN 16094810 Ki = 100 nM T28893 CTYI57 16115796 Ki = 0.7586 nM T28893 C5HSD9 16115797 Ki = 0.3467 nM T28893 CQ85FK 16115798 Ki = 1.479 nM T28893 CR1Z4N 16115799 Ki = 0.912 nM T28893 CLA6E0 16115800 Ki = 2.344 nM T28893 CTE0R7 16115942 Ki = 0.955 nM T28893 C7IC9E 16115944 Ki = 0.2512 nM T28893 CQ3C9X 16115946 Ki = 0.5012 nM T28893 C0JGY1 16115950 Ki = 3.467 nM T28893 CZ67DO 16115951 Ki = 1.38 nM T28893 CO3YU4 16116082 Ki = 0.2951 nM T28893 C3IKJ0 16116084 Ki = 0.1175 nM T28893 CWU6P3 16123945 EC50 = 5.012 nM T28893 CZ2IS9 16660294 Ki > 10000 nM T28893 CO1W8M 16721019 Ki = 18 nM T28893 CGCY91 16742745 IC50 = 1030 nM T28893 C2IJ3D 16742746 IC50 = 962 nM T28893 C4URY2 16742747 IC50 > 10000 nM T28893 C8V1KM 16745235 IC50 = 325 nM T28893 CDB83R 17516658 EC50 > 30000 nM T28893 C45VOE 18342968 Ki = 242 nM T28893 C5CKH8 18920309 IC50 = 141.25 nM T28893 CE93IQ 18920330 IC50 = 0.004 nM T28893 CIUC68 18920353 IC50 = 9 nM T28893 CD6G2M 19612616 IC50 = 3801.89 nM T28893 C7T8JC 19958494 Ki > 10000 nM T28893 C6LI5E 19958507 Ki > 10000 nM T28893 CBO56R 20449980 EC50 = 317 nM T28893 CVJS49 20918651 EC50 = 776.25 nM T28893 C61NXP 20918653 EC50 = 1000 nM T28893 CD0L9F 21262774 EC50 = 537.03 nM T28893 C3T5HF 21509921 Ki = 3981.07 nM T28893 C4FNZ8 21862266 Ki = 2900 nM T28893 C3SXF7 21947646 IC50 = 862 nM T28893 CKW4S9 22730942 EC50 = 1.9 nM T28893 C5WCD3 22745278 EC50 = 2.1 nM T28893 C3IQT5 23352279 Ki = 480 nM T28893 C5SUY3 23352285 Ki = 990 nM T28893 CC29GD 23633277 IC50 > 10000 nM T28893 C1RV7P 23633348 IC50 > 10000 nM T28893 CU1LK3 23633350 IC50 > 10000 nM T28893 CKN67W 23633553 IC50 > 10000 nM T28893 CG37EL 23633557 IC50 > 10000 nM T28893 C5U3NL 23633697 IC50 > 10000 nM T28893 CVC80Z 23633837 IC50 > 10000 nM T28893 C8P9GL 23633839 IC50 > 10000 nM T28893 C5UVZ9 23634061 IC50 > 10000 nM T28893 C5ZF2X 23634210 IC50 > 10000 nM T28893 C4KW2T 23634279 IC50 > 10000 nM T28893 CVF78O 23634281 IC50 > 10000 nM T28893 C5Y1MK 23983764 Ki = 91.2 nM T28893 CEVA58 24121307 IC50 = 1000 nM T28893 CL4WV2 24180125 IC50 = 8020 nM T28893 CXCO68 24192587 Ki = 85.7 nM T28893 CBXC05 24424330 IC50 = 22 nM T28893 C8KTP0 24739387 IC50 > 10000 nM T28893 C70CVK 24739554 IC50 = 8900 nM T28893 CSDA50 24739886 IC50 = 5000 nM T28893 CKVQ51 24749924 IC50 = 25 nM T28893 CCW9N3 24749925 IC50 = 5 nM T28893 CXNY61 24749926 IC50 = 6161 nM T28893 C7I4LK 24750278 IC50 = 50 nM T28893 CT21RV 24750279 IC50 = 26 nM T28893 C5TIP2 24750281 IC50 = 1129 nM T28893 CI6JQ2 24751745 EC50 = 1.778 nM T28893 CY21RE 24841480 Ki = 2 nM T28893 C4SY8G 24846938 Ki = 1.32 nM T28893 C7ZEF0 24856058 IC50 = 1425 nM T28893 CF26NI 24865894 Ki = 12882.5 nM T28893 CJ4FM6 24865895 Ki = 8317.64 nM T28893 C3C0KP 24894134 EC50 > 50000 nM T28893 C9YN3A 24894514 Ki = 43651.58 nM T28893 C8ND1U 24894515 Ki = 77624.71 nM T28893 CX2HR8 24894516 Ki = 36307.81 nM T28893 CG4B9R 24894624 Ki = 30902.95 nM T28893 C7KF9R 24894626 Ki = 5623.41 nM T28893 CFA60S 24894627 Ki = 5248.07 nM T28893 CT8B3K 24894629 Ki = 7413.1 nM T28893 CMF04K 24894631 Ki = 33113.11 nM T28893 CP08SJ 24894632 Ki = 26915.35 nM T28893 CLJK58 24894633 Ki = 44668.36 nM T28893 CR86FA 24894634 Ki = 51286.14 nM T28893 C9J3NX 24894636 Ki = 13803.84 nM T28893 CUY89J 24936155 Ki = 230 nM T28893 C1LKN4 24964946 EC50 = 270 nM T28893 CK78TS 24965292 EC50 = 380 nM T28893 CICV53 24965294 EC50 = 84 nM T28893 CQ3ER0 24967069 EC50 = 41 nM T28893 CR7D1L 24967746 EC50 = 0.3981 nM T28893 C5MYC3 25010776 EC50 = 2300 nM T28893 C1VRJ3 25014630 IC50 = 8600 nM T28893 C18VYH 25015647 EC50 > 40000 nM T28893 CP6K8J 25024727 IC50 > 10000 nM T28893 CA20NZ 25025581 Ki = 158.49 nM T28893 C8JW9U 25034110 IC50 = 12589.25 nM T28893 C9OC1I 25034111 IC50 = 1000 nM T28893 C3DB4P 25034112 IC50 = 19952.62 nM T28893 CH67WY 25034180 IC50 = 3981.07 nM T28893 C2G1JK 25053351 Ki = 11 nM T28893 CBY3O2 25070582 IC50 = 300 nM T28893 CXBF68 25110764 EC50 = 0.85 nM T28893 C50IKG 25110765 EC50 = 0.76 nM T28893 CK0BT7 25147647 Ki = 2290.87 nM T28893 CGH08V 25164128 IC50 = 630.96 nM T28893 CE2OG1 25199525 EC50 = 25.12 nM T28893 CRFJ43 25207745 EC50 = 10 nM T28893 CP2T6G 25230693 EC50 = 2.512 nM T28893 C45ZNS 42596928 Ki = 0.7943 nM T28893 C5DC7E 42598357 EC50 = 3.162 nM T28893 CO6QB0 42598358 EC50 = 1 nM T28893 CDPA93 42598359 EC50 = 12.59 nM T28893 CAM5P6 42598360 EC50 = 2.512 nM T28893 C58SRK 42598586 EC50 = 199.53 nM T28893 CYL45Z 42598591 EC50 = 0.5012 nM T28893 C6S2HI 42598828 EC50 = 1.259 nM T28893 C2GYA4 42598829 EC50 = 7.943 nM T28893 C5CZ7P 42599068 EC50 = 3.162 nM T28893 C7O2ZV 42599070 EC50 = 0.3981 nM T28893 C6BUZ5 42599071 EC50 = 2.512 nM T28893 CMX21F 42601144 IC50 > 10000 nM T28893 CS40ML 44123747 IC50 > 10000 nM T28893 CM5XL8 44186798 EC50 = 48 nM T28893 CMR7T1 44204999 EC50 = 398.11 nM T28893 C2XZP8 44206730 EC50 = 130 nM T28893 COT2Z0 44206959 EC50 = 46 nM T28893 CY5JI9 44207208 EC50 = 100 nM T28893 CW04VH 44207445 EC50 = 310 nM T28893 C4TW7Z 44207447 EC50 = 20 nM T28893 CS17PI 44207904 EC50 = 19 nM T28893 CY8J9L 44207907 EC50 = 180 nM T28893 C2HRX1 44207908 EC50 = 110 nM T28893 C9T0PX 44208358 EC50 = 86 nM T28893 C6GXL0 44208359 EC50 = 13 nM T28893 CQ61TP 44208564 EC50 = 15 nM T28893 CV1P7W 44213237 Ki = 30 nM T28893 C47KIQ 44213238 Ki = 292 nM T28893 CY1ZK0 44213239 Ki = 30 nM T28893 CGCX24 44214356 EC50 = 258.9 nM T28893 CX54AP 44215433 EC50 = 160 nM T28893 CPW7K9 44232679 IC50 = 0.34 nM T28893 CU2T6F 44232680 IC50 = 0.6 nM T28893 CEQO63 44232682 IC50 = 0.31 nM T28893 CW1V2M 44232684 IC50 = 0.38 nM T28893 CDRG51 44232927 IC50 = 0.2 nM T28893 CVQB56 44232930 IC50 = 0.2 nM T28893 C4MK8P 44232931 IC50 = 0.19 nM T28893 CU6Q8I 44232952 Ki = 0.1 nM T28893 C91ZIE 44232953 IC50 = 1276 nM T28893 C4OK7Y 44233172 IC50 = 0.23 nM T28893 C4Y3XC 44233174 IC50 = 1.12 nM T28893 CYC26A 44233176 IC50 = 0.28 nM T28893 C6WXJ9 44233187 IC50 = 770 nM T28893 CQM1T9 44233189 IC50 = 277 nM T28893 CAHP03 44233190 Ki = 1 nM T28893 CA59KP 44233191 Ki = 1.259 nM T28893 C8LM6H 44233399 Ki = 0.08 nM T28893 CCK0D4 44233400 IC50 = 0.23 nM T28893 C3OY7U 44233402 IC50 = 0.16 nM T28893 CP1G4K 44233417 IC50 = 1017 nM T28893 CA7LB8 44233419 IC50 = 2198 nM T28893 C5Q3EJ 44233675 IC50 = 105 nM T28893 CHK5U6 44233928 IC50 = 596 nM T28893 C9OG5Z 44234194 IC50 = 1597 nM T28893 CX21NW 44235638 IC50 = 15 nM T28893 C17PIF 44235871 IC50 = 0.26 nM T28893 CBU6A0 44236098 IC50 = 0.23 nM T28893 CK0JC2 44236099 IC50 = 0.24 nM T28893 CUD0K2 44236100 IC50 = 0.29 nM T28893 CG13KU 44236331 IC50 = 0.63 nM T28893 CH12JO 44236333 IC50 = 1.26 nM T28893 C73FXN 44236335 IC50 = 0.43 nM T28893 CR8WZ1 44236337 IC50 = 100 nM T28893 CA15LQ 44236339 IC50 = 0.29 nM T28893 C9JGH5 44247476 IC50 = 2000 nM T28893 CN7QV2 44247479 IC50 > 10000 nM T28893 CX7L4D 44247481 IC50 > 10000 nM T28893 C5UAT0 44247486 IC50 = 320 nM T28893 C37BFM 44247488 IC50 = 1100 nM T28893 C54CHX 44247490 IC50 = 2600 nM T28893 CDLJ56 44247492 IC50 = 4500 nM T28893 C8LN7D 44247495 IC50 > 10000 nM T28893 C2QIA0 44247496 IC50 > 10000 nM T28893 CPYC57 44247497 IC50 > 10000 nM T28893 C3Q0SZ 44247502 IC50 > 10000 nM T28893 C86ENQ 44247504 IC50 > 10000 nM T28893 COS20B 44247505 IC50 > 10000 nM T28893 C3JAL1 44247512 IC50 > 10000 nM T28893 C7K0JL 44247513 IC50 > 10000 nM T28893 CG8L7X 44247523 IC50 > 10000 nM T28893 C7MY2N 44247806 Ki = 20000 nM T28893 CF9TE1 44247935 Ki = 0.32 nM T28893 C85DHY 44250284 Ki = 4800 nM T28893 CE2V4Z 44251554 EC50 = 2300 nM T28893 CT6N4S 44251555 EC50 = 860 nM T28893 CGR6J0 44251556 EC50 = 600 nM T28893 C0K9BZ 44251557 EC50 = 2300 nM T28893 CW02TZ 44251558 EC50 = 1100 nM T28893 CS2DH6 44251559 EC50 = 1200 nM T28893 C2K0VZ 44253016 EC50 = 12.59 nM T28893 C2LFH7 44274302 Ki = 7079.46 nM T28893 CZX4M3 44274317 Ki = 26915.35 nM T28893 C5L3FV 44274400 Ki = 28183.83 nM T28893 CF47ZS 44274417 Ki = 21877.62 nM T28893 CCK63Z 44274432 Ki = 48977.88 nM T28893 CZ1U0E 44274433 Ki = 23988.33 nM T28893 C3XP7C 44274441 Ki = 11481.54 nM T28893 CO1RL0 44274468 Ki = 18620.87 nM T28893 C9JX7D 44274469 Ki = 9549.93 nM T28893 CF36IC 44274477 Ki = 29512.09 nM T28893 CE20CZ 44275807 Ki = 1621.81 nM T28893 CC2OD4 44278111 Ki > 10000 nM T28893 CRMA84 44278114 Ki > 10000 nM T28893 CF0Y4M 44278115 Ki > 10000 nM T28893 CFS16C 44285542 Ki = 6500 nM T28893 CSP92A 44285557 Ki = 15000 nM T28893 CR6D5Q 44285558 Ki = 20000 nM T28893 CXB29F 44285864 Ki = 6300 nM T28893 CCN0Q7 44299323 Ki = 14 nM T28893 CSB7T8 44299324 Ki = 22 nM T28893 C07GVY 44299328 Ki = 75 nM T28893 CUD8P0 44299369 Ki = 690 nM T28893 C1GX3I 44299477 Ki = 2500 nM T28893 C9Z0LT 44299564 Ki = 2570.4 nM T28893 CX28HR 44299589 Ki = 2344.23 nM T28893 CPL36O 44299599 Ki = 3235.94 nM T28893 CFN95A 44299616 Ki = 1513.56 nM T28893 CE4L1V 44299635 Ki = 5370.32 nM T28893 C9TWN3 44302727 IC50 = 9017.8 nM T28893 C5S8UL 44302728 IC50 = 12903.4 nM T28893 CQ4B5T 44302741 IC50 = 1961.9 nM T28893 C0AZF5 44302755 IC50 = 8221.3 nM T28893 CR5T1J 44302775 IC50 = 4250 nM T28893 CY8PD1 44302776 IC50 = 3277.5 nM T28893 C7GY5J 44302788 IC50 = 3788 nM T28893 CAV72D 44302793 IC50 = 32653.5 nM T28893 CV9QM6 44302813 IC50 = 5009.3 nM T28893 C43QTF 44302833 IC50 = 6109.7 nM T28893 CF74EQ 44302834 IC50 = 1959.3 nM T28893 C6J3EY 44302879 IC50 = 7121.2 nM T28893 CIU20B 44302900 IC50 = 4058 nM T28893 CGNA91 44302901 IC50 = 10766.6 nM T28893 CY47SI 44303018 EC50 = 10.5 nM T28893 C6H2ZT 44303019 EC50 = 71 nM T28893 C6BMW2 44303286 EC50 = 70.5 nM T28893 C3L8RU 44303293 EC50 = 1810 nM T28893 C0SLC4 44303294 EC50 = 46 nM T28893 C7X1GV 44303314 EC50 = 2.5 nM T28893 C85QFH 44303323 EC50 = 4.5 nM T28893 C7J1HZ 44303327 EC50 = 61.9 nM T28893 CD9A5N 44303396 EC50 = 107 nM T28893 CW6O3V 44303397 EC50 = 9 nM T28893 C5VJK4 44303408 EC50 = 110 nM T28893 C9TUK2 44303424 EC50 = 1200 nM T28893 C03MFZ 44308733 Ki = 1.5 nM T28893 CT3V7Z 44308746 Ki = 4.7 nM T28893 C0Z3JQ 44308798 Ki = 1900 nM T28893 CN9M6A 44308799 Ki = 760 nM T28893 C38WIK 44308809 Ki = 55 nM T28893 CF06ON 44308818 Ki = 210 nM T28893 C90FZB 44308831 Ki = 140 nM T28893 CK14IH 44308832 Ki = 1.3 nM T28893 COE23J 44308861 Ki = 1.8 nM T28893 CMX10C 44308899 Ki = 2.1 nM T28893 CN5G8U 44308900 Ki = 11 nM T28893 CLJ71S 44308910 Ki = 30 nM T28893 C3L7HC 44308912 Ki = 2.1 nM T28893 CP0G8R 44308913 Ki = 21 nM T28893 CY6TU4 44309089 Ki = 23 nM T28893 CMAC70 44309090 Ki = 140 nM T28893 CND98T 44309107 Ki = 740 nM T28893 CEFY94 44309108 Ki = 630 nM T28893 C61LZX 44309135 Ki = 140 nM T28893 CY8D9F 44309151 Ki = 92 nM T28893 CD7QT6 44309153 Ki = 11 nM T28893 C7CQ3N 44309208 Ki = 14 nM T28893 C3B0IJ 44309209 Ki = 37 nM T28893 CIG89A 44309231 Ki = 1 nM T28893 CSW73I 44311704 Ki = 116.68 nM T28893 C2R3SX 44311716 Ki = 33.34 nM T28893 CJ9C3I 44311717 Ki = 37.41 nM T28893 C7QD0Y 44311718 Ki = 57.02 nM T28893 CH7IJ2 44311760 Ki = 42 nM T28893 CGY95E 44311761 Ki = 60.81 nM T28893 CT41MZ 44311762 Ki = 9.099 nM T28893 CT6Y9V 44311771 Ki = 25.7 nM T28893 CJ3F7Y 44311784 Ki = 9.795 nM T28893 CO28DW 44311785 Ki = 40.74 nM T28893 CI2LP0 44311786 Ki = 60.39 nM T28893 CV52TA 44311823 Ki = 10.79 nM T28893 CQ51WZ 44311835 Ki = 95.72 nM T28893 CT8U1D 44311987 Ki = 74.47 nM T28893 CSA8M2 44312007 Ki = 10.5 nM T28893 C4ENG6 44312024 Ki = 14.76 nM T28893 CBE37N 44312066 Ki = 52 nM T28893 C7W3FI 44312081 Ki = 57 nM T28893 C6OP9A 44312083 Ki = 11 nM T28893 COX3S1 44312132 Ki = 4770 nM T28893 C89QFR 44312152 Ki = 77 nM T28893 CZ65YU 44312450 Ki = 8 nM T28893 C6YGO9 44312451 Ki = 6 nM T28893 CZ84YU 44312455 Ki = 106 nM T28893 CWN9H1 44312460 Ki = 96 nM T28893 CL6M1O 44312464 Ki = 85 nM T28893 CP4S2D 44312468 Ki = 200 nM T28893 CM0Z7K 44313166 Ki = 3110 nM T28893 CU9FV1 44313489 Ki = 581 nM T28893 CC5W6M 44313626 Ki = 63 nM T28893 C04VNU 44313630 Ki = 20 nM T28893 C71NXG 44313631 Ki > 10000 nM T28893 CVX13Q 44318736 Ki = 29 nM T28893 CT58BQ 44318766 Ki = 970 nM T28893 CR2T3J 44318817 Ki = 230 nM T28893 CL0HY5 44318929 Ki = 1000 nM T28893 C01CVA 44318930 Ki = 450 nM T28893 CGSU92 44326538 Ki = 166 nM T28893 C8RGU2 44327038 IC50 = 247 nM T28893 C7MRA5 44327263 IC50 = 250 nM T28893 C39VCG 44327295 IC50 = 1228 nM T28893 C9TOB0 44327400 IC50 = 806 nM T28893 C8HF1K 44327401 IC50 > 10 nM T28893 C8VE3G 44327424 IC50 = 260 nM T28893 CSE35C 44328347 Ki = 2040 nM T28893 CM6D4U 44328348 Ki > 5000 nM T28893 CX4M2I 44328356 Ki > 8000 nM T28893 C8O4PB 44328540 Ki = 330 nM T28893 CTX68J 44328560 Ki >> 200 nM T28893 CP5W3M 44328561 Ki = 422 nM T28893 CO18HJ 44329977 EC50 = 0.99 nM T28893 CDC01L 44330073 EC50 > 100 nM T28893 CYC95E 44330074 EC50 = 1 nM T28893 CL5EU8 44330080 EC50 = 28.3 nM T28893 CBTX60 44330081 EC50 = 0.5 nM T28893 C1BXQ3 44330323 IC50 = 144.54 nM T28893 CD9ZS8 44342270 IC50 = 1780 nM T28893 CSK4B0 44346542 IC50 = 27.3 nM T28893 C1A2OH 44350993 EC50 = 22.3 nM T28893 C27ELM 44350994 EC50 = 430.9 nM T28893 CR0VU2 44351073 EC50 = 225 nM T28893 C6IQF4 44351242 EC50 = 1 nM T28893 CU2X1V 44356367 IC50 = 13000 nM T28893 CXJ4G7 44364174 Ki = 88 nM T28893 C3VT2M 44379080 Ki = 129 nM T28893 CU68GE 44379281 Ki = 70 nM T28893 CUA24S 44379508 Ki = 67.1 nM T28893 CG85AM 44380820 Ki = 510 nM T28893 CQ7P3Y 44382840 Ki = 601 nM T28893 CCYU52 44382841 Ki = 179 nM T28893 CW2J6Y 44382858 Ki = 427 nM T28893 C7VOM3 44382864 Ki > 900 nM T28893 CKC6L3 44382865 Ki = 416 nM T28893 C8OZ2J 44382880 Ki = 353 nM T28893 C3TX9A 44382974 Ki = 464 nM T28893 C5JHQ8 44383064 Ki = 304 nM T28893 C26DNS 44383065 Ki = 136 nM T28893 CO3UJ2 44383238 Ki = 38 nM T28893 C61QNW 44383352 Ki = 312 nM T28893 C0G2RO 44383373 Ki = 579 nM T28893 CXG5Q3 44383489 Ki = 445 nM T28893 C1BP8Z 44383490 Ki = 1361 nM T28893 C9T1BR 44383492 Ki = 581 nM T28893 CG90DX 44383554 Ki = 376 nM T28893 CA8T0K 44383595 Ki = 341 nM T28893 CDA8W1 44383613 Ki = 857 nM T28893 C5X3RM 44383653 Ki = 4.3 nM T28893 CZ8E1C 44383766 Ki > 420 nM T28893 CY6B5S 44384258 Ki = 399 nM T28893 C36YBR 44384326 Ki = 554 nM T28893 CIDW56 44384327 Ki = 1533 nM T28893 C7YTV9 44385809 Ki = 300 nM T28893 CHD9O7 44386115 Ki = 77 nM T28893 C2VN8S 44392087 IC50 = 400 nM T28893 CG2VT0 44392899 Ki > 1400 nM T28893 CFY5B7 44392905 Ki = 790 nM T28893 CIW3F6 44392933 Ki = 68 nM T28893 C1GB6S 44392936 Ki > 1400 nM T28893 CCX9A6 44392956 Ki > 1400 nM T28893 C2H4QG 44392960 Ki = 418 nM T28893 C0HP4R 44392966 Ki = 122 nM T28893 C3MKY5 44392967 Ki = 811 nM T28893 CPVS57 44392974 Ki = 177 nM T28893 CD5PS0 44392978 Ki = 640 nM T28893 CS8F0W 44392983 Ki = 446 nM T28893 C53TYX 44396257 Ki = 69.7 nM T28893 CALU25 44396260 Ki = 53.5 nM T28893 CB6E7U 44396263 Ki = 135 nM T28893 C1UN8C 44396277 Ki > 1000 nM T28893 C1B4QL 44403095 Ki > 10000 nM T28893 C1YL7Z 44403098 Ki > 10000 nM T28893 CFV98A 44403101 Ki > 10000 nM T28893 C6OY9S 44403102 Ki > 10000 nM T28893 CH4SX6 44403105 Ki > 10000 nM T28893 C12FIH 44403106 Ki > 10000 nM T28893 C4LKC1 44404394 Ki > 10000 nM T28893 C3EJ4G 44404396 Ki > 10000 nM T28893 C6GLV1 44408714 Ki = 1949.84 nM T28893 C4QTI3 44415886 Ki = 800 nM T28893 CC9AV3 44418764 Ki = 199.53 nM T28893 CV6UQ3 44419370 Ki > 100000 nM T28893 C2N5LX 44422691 Ki = 30199.52 nM T28893 CIRB78 44422696 Ki = 74131.02 nM T28893 CHT24X 44422698 Ki < 100000 nM T28893 CDE8A1 44428745 Ki = 19.95 nM T28893 CRN6M1 44431367 Ki = 220 nM T28893 CQD71K 44431369 Ki = 220 nM T28893 CAE86V 44431370 Ki = 260 nM T28893 C92HNF 44431372 Ki = 200 nM T28893 CI36TZ 44431375 Ki = 540 nM T28893 CZ12VG 44431376 Ki = 380 nM T28893 CS0H4C 44431380 Ki = 31 nM T28893 C5FJR6 44431381 Ki = 21 nM T28893 CG0BM9 44431382 Ki = 18 nM T28893 CW60PY 44431383 Ki = 12 nM T28893 C0JL9K 44431384 Ki = 5.9 nM T28893 C3S0AU 44431386 Ki = 86 nM T28893 C0T5AL 44431387 Ki = 52 nM T28893 C15WZI 44431388 Ki = 140 nM T28893 C29VWS 44431389 Ki = 19 nM T28893 C1LJ6G 44431391 Ki = 36 nM T28893 CLA76R 44431393 Ki = 1.8 nM T28893 C53UEG 44434115 IC50 = 518 nM T28893 CG45PO 44437242 Ki > 10000 nM T28893 C6I2JO 44437248 Ki = 7680 nM T28893 CZI05O 44437258 Ki = 3376 nM T28893 C7VP1Y 44437297 Ki = 7367 nM T28893 C5GT7C 44437302 Ki > 10000 nM T28893 C37QFT 44437307 Ki = 6958 nM T28893 C36LXN 44446840 Ki < 100000 nM T28893 C4IXY7 44448987 IC50 > 5000 nM T28893 COP51N 44448988 IC50 > 5000 nM T28893 CUM32L 44449149 IC50 = 93 nM T28893 CR4ZT2 44450620 Ki = 19054.61 nM T28893 C5H7OQ 44450621 Ki = 14125.38 nM T28893 CZ50IM 44450622 Ki = 5888.44 nM T28893 CS5CD3 44450624 Ki = 8317.64 nM T28893 CFN4B5 44450637 Ki = 21379.62 nM T28893 C12XGE 44456400 Ki > 10000 nM T28893 CD58GR 44456521 IC50 = 7079.46 nM T28893 C83YOC 44456549 IC50 = 3981.07 nM T28893 CC6UO5 44456576 IC50 = 1905.46 nM T28893 CZRF79 44456577 IC50 = 77624.71 nM T28893 CF9C3L 44456598 IC50 = 1000 nM T28893 CH1MK7 44456600 IC50 = 162.18 nM T28893 C3PO1X 44456623 IC50 = 309.03 nM T28893 CWMX31 44456645 IC50 = 1071.52 nM T28893 CN64CM 44456845 IC50 = 58.88 nM T28893 C2VT7Z 44456846 IC50 = 616.6 nM T28893 CT8UN7 44456863 IC50 = 870.96 nM T28893 C60UTA 44456864 IC50 = 275.42 nM T28893 CQ0WM7 44469273 IC50 > 5000 nM T28893 C4DL5C 44469677 IC50 > 10000 nM T28893 CVA67X 44568347 Ki = 64 nM T28893 CY9C2A 44571572 Ki > 100000 nM T28893 CM0D1J 44575653 IC50 = 7 nM T28893 CN68YI 44578707 Ki = 1445.44 nM T28893 CHUN40 44578928 EC50 = 1500 nM T28893 CZYP06 44578975 EC50 = 1800 nM T28893 CCIT12 44578976 EC50 = 120 nM T28893 CW53ZF 44578977 EC50 = 1100 nM T28893 CYHM34 44578978 EC50 = 490 nM T28893 CGF7A4 44579375 EC50 = 1030 nM T28893 C1OCB6 44579416 EC50 = 1600 nM T28893 CARW17 44579417 EC50 = 356 nM T28893 C2DFV7 44579418 EC50 = 1.06 nM T28893 CTC8H6 44579419 EC50 = 1.71 nM T28893 CYR0O3 44579457 EC50 = 1.04 nM T28893 CF1EA4 44579458 EC50 > 10 nM T28893 C6HMP4 44589495 IC50 = 1000 nM T28893 C9U3KY 44589496 IC50 = 1000 nM T28893 CXL82E 44589497 IC50 > 3162.28 nM T28893 CLGW57 44589498 IC50 = 1000 nM T28893 C1KY5I 44589499 IC50 > 3162.28 nM T28893 CM2JG4 44589500 EC50 = 11100 nM T28893 CX3ZW4 44589501 EC50 = 930 nM T28893 C6H0WS 44589502 EC50 = 7110 nM T28893 CSE54A 44589503 EC50 = 1400 nM T28893 C0N4QF 44589529 IC50 > 3162.28 nM T28893 CQ4Y8O 44589531 EC50 = 6500 nM T28893 COE0T7 44589569 IC50 > 3162.28 nM T28893 CE4FX5 44589570 IC50 > 3162.28 nM T28893 C9J2RO 44589571 IC50 > 3162.28 nM T28893 CKY4F8 44589572 IC50 > 3162.28 nM T28893 CX19BO 44589573 IC50 > 3162.28 nM T28893 C10LXB 44589574 IC50 > 3162.28 nM T28893 CUD4M8 44589575 IC50 > 3162.28 nM T28893 CL40CM 44589593 EC50 = 2600 nM T28893 CKS5V4 44589594 EC50 = 2300 nM T28893 CXB30W 44589595 EC50 = 3300 nM T28893 CM5LJ8 44589596 EC50 = 4100 nM T28893 CPXE19 44589643 EC50 = 4400 nM T28893 C8AJO6 44589644 EC50 > 10000 nM T28893 CFS1A4 44589645 EC50 = 9600 nM T28893 C71EHI 44589646 EC50 = 3600 nM T28893 CQB5A9 44589681 EC50 = 2100 nM T28893 CE06LX 44589984 IC50 = 794.33 nM T28893 C6LC7V 44590033 IC50 = 501.19 nM T28893 CL57OY 44590034 IC50 = 2511.89 nM T28893 CO3GX2 44590035 IC50 = 1000 nM T28893 CT58OX 44590036 IC50 = 1000 nM T28893 C2H9IW 44590122 IC50 = 251.19 nM T28893 CJ2M0R 44590123 IC50 = 1258.93 nM T28893 C5JVF6 44590124 IC50 > 3162.28 nM T28893 C3G5LY 44590125 IC50 = 1995.26 nM T28893 CF4DI1 44590166 IC50 > 3162.28 nM T28893 CYC47W 44590167 IC50 = 630.96 nM T28893 CH61KJ 44590182 IC50 = 1000 nM T28893 C1Q6SJ 44590186 EC50 = 2710 nM T28893 CF6E4J 44590187 EC50 = 510 nM T28893 CL7V4S 44590188 EC50 = 2110 nM T28893 CA30UF 44590189 EC50 = 910 nM T28893 CUA62X 44593616 Ki = 74.13 nM T28893 CN9ID8 44593617 Ki = 109.65 nM T28893 CDM56I 44593618 Ki = 14.13 nM T28893 CU63PQ 44593619 Ki = 10 nM T28893 CL8D2S 44593620 Ki = 38.02 nM T28893 CI97KQ 44593621 Ki = 93.33 nM T28893 CNZ1U7 44593651 IC50 < 1 nM T28893 CL5O8E 44602489 EC50 > 30000 nM T28893 CH2Z3O 44610056 Ki = 0.16 nM T28893 CVZ6Y1 44627739 Ki = 35.48 nM T28893 CE6A9F 44627740 Ki = 1.23 nM T28893 C6EU7P 44627741 Ki = 42.66 nM T28893 CW40TR 44627742 Ki = 13.49 nM T28893 C5GIU6 44627743 Ki = 23.44 nM T28893 CK9DO1 44627745 Ki = 2.089 nM T28893 CJ8S1L 44627747 Ki = 11.48 nM T28893 C5LY8C 44627851 Ki = 6.607 nM T28893 CC4A3X 44627853 Ki = 1.23 nM T28893 CH4N5J 44627854 Ki = 22.91 nM T28893 CO8C6D 44627855 Ki = 190.55 nM T28893 COL8E1 44627856 Ki = 1230.27 nM T28893 C6WS7M 44627857 Ki = 0.6918 nM T28893 C43BJY 44627859 Ki = 9.12 nM T28893 CW0X6A 44627955 Ki = 47.86 nM T28893 CXNF31 44627957 Ki = 331.13 nM T28893 C2R8DF 44768972 IC50 > 10000 nM T28893 C9U0VH 45259185 Ki = 53.7 nM T28893 CNC1R2 45259186 Ki = 15.85 nM T28893 CP2CZ7 45259187 Ki = 56.23 nM T28893 CW14TS 45259188 Ki = 3.02 nM T28893 CO8W1X 45259189 Ki = 6.918 nM T28893 CF16YZ 45259190 Ki = 19.5 nM T28893 C1K0ZH 45259193 Ki = 0.3162 nM T28893 CQGM36 45262105 Ki = 630.96 nM T28893 C7L1CU 45266348 Ki = 21.88 nM T28893 CK8N4L 45266386 Ki = 93325.43 nM T28893 CJQ8C6 45266387 IC50 = 12.59 nM T28893 C2IV6N 45266389 IC50 = 31.62 nM T28893 C7WBU9 45266390 IC50 = 100 nM T28893 C5J2TE 45266397 IC50 = 251.19 nM T28893 C0O9TA 45266401 IC50 = 39.81 nM T28893 C5P1NR 45266404 IC50 = 1995.26 nM T28893 CJ9W5C 45266406 IC50 = 158.49 nM T28893 CH74XR 45266408 IC50 = 25.12 nM T28893 CGH8T0 45266411 IC50 = 630.96 nM T28893 C73TVO 45266437 IC50 = 100 nM T28893 C5PTZ9 45266459 IC50 = 79.43 nM T28893 C0D4LK 45266462 IC50 = 1258.93 nM T28893 CUK8N1 45266464 IC50 = 251.19 nM T28893 CRI98L 45266467 IC50 = 199.53 nM T28893 C0AV6F 45266469 IC50 = 100 nM T28893 CZA73U 45266470 IC50 = 10 nM T28893 C0FHW1 45266476 IC50 = 50.12 nM T28893 CZ23VF 45266478 IC50 = 39.81 nM T28893 C6SV5O 45267774 Ki > 10000 nM T28893 CHQ05B 45267775 IC50 > 10000 nM T28893 C65LBY 45268662 Ki = 89 nM T28893 CCFG82 45269436 IC50 = 14747 nM T28893 CFZ01K 45270350 IC50 = 3860 nM T28893 CW6HL5 45271167 Ki = 3581 nM T28893 CA0SD1 45272895 Ki > 10000 nM T28893 CE71LQ 45273833 Ki = 2745 nM T28893 C3QU2C 45487384 IC50 > 5000 nM T28893 CK6X3B 45786849 Ki = 10000 nM T28893 CL0M1G 46174144 Ki = 0.05 nM T28893 CU4V5R 46227410 Ki > 100000 nM T28893 CWQ1L9 46227412 Ki = 24547.09 nM T28893 CX2E6A 46227414 Ki > 100000 nM T28893 C0Z4RD 46227416 Ki > 100000 nM T28893 CK2R5G 46227454 Ki > 100000 nM T28893 C8OZI6 46227456 Ki = 47863.01 nM T28893 CB45NM 46227458 Ki > 100000 nM T28893 C1J0IF 46227460 Ki = 67608.3 nM T28893 CQ4DI6 46227480 Ki = 95499.26 nM T28893 CHKL80 46227482 Ki = 19952.62 nM T28893 CVP7T6 46227484 Ki = 38018.94 nM T28893 CC6RH5 46227486 Ki > 100000 nM T28893 CSQ0V3 46227554 Ki > 100000 nM T28893 CC68WI 46830289 Ki > 10000000 nM T28893 CK1X9S 46830361 IC50 = 350 nM T28893 C1Q0MH 46830362 IC50 = 490 nM T28893 CH3ID7 46830363 IC50 = 2600 nM T28893 CH83EL 46854806 Ki = 350 nM T28893 CP6DN0 46861858 Ki = 40 nM T28893 CW1FS9 46861860 Ki = 2900 nM T28893 C2QH7O 46865650 Ki = 3700 nM T28893 CC5KR7 46865978 Ki > 10000 nM T28893 C01YTE 46871665 EC50 = 10 nM T28893 CUY51M 46871666 EC50 = 19.95 nM T28893 CYLZ50 46871844 EC50 = 0.7943 nM T28893 CCZ5I8 46883796 IC50 = 2900 nM T28893 CVCF68 46883843 IC50 = 4700 nM T28893 CW6A9I 46884062 IC50 = 3700 nM T28893 C04JMO 46884063 Ki > 10000 nM T28893 CR1Z8E 46884119 Ki > 10000 nM T28893 CR0CQ9 46884120 Ki > 10000 nM T28893 C9OYT5 46884152 Ki = 2200 nM T28893 CCI32B 46884153 Ki > 10000 nM T28893 C2JQE7 46884154 Ki > 10000 nM T28893 C20HET 46884155 Ki > 10000 nM T28893 C0HYN3 46884200 Ki > 10000 nM T28893 CM6A8S 46884201 Ki = 4759000 nM T28893 CW94IK 46884202 Ki > 10000000 nM T28893 COPQ16 46884600 Ki > 10000 nM T28893 C85MOA 46884637 Ki > 10000 nM T28893 C36NKV 46884638 Ki > 10000 nM T28893 CQ84IF 46884639 Ki = 15000 nM T28893 CZGS15 46884640 Ki = 17000 nM T28893 CZ72SW 46884641 Ki > 10000 nM T28893 CA3Z6G 46884666 Ki = 2400 nM T28893 C8DBY0 46884667 Ki = 3600 nM T28893 CU3BG6 46884668 Ki > 10000 nM T28893 CPG14Q 46884669 Ki > 10000 nM T28893 C7R9AK 46884670 Ki > 10000 nM T28893 C64KNW 46884698 Ki = 2000 nM T28893 C0ASK4 46884699 Ki > 10000 nM T28893 CYNU85 46884731 Ki > 10000 nM T28893 CJ6O8D 46884732 Ki > 10000 nM T28893 C9QT7G 46884733 Ki > 10000 nM T28893 CL6Z7Q 46884734 Ki > 10000 nM T28893 C6PRX8 46884735 Ki = 3500 nM T28893 CWK8I4 46884736 Ki > 10000 nM T28893 CJK1Z5 46888857 Ki = 2800 nM T28893 CX92WH 46889257 Ki = 2500 nM T28893 C01DMO 46889258 Ki = 1500 nM T28893 CAY6U8 46890714 EC50 = 100 nM T28893 C08IDT 46890715 EC50 = 63.1 nM T28893 C1M0LP 46890716 EC50 > 10000 nM T28893 CS6JV9 46890717 EC50 = 158.49 nM T28893 C83ILZ 46890718 EC50 = 1000 nM T28893 CW1DM2 46890719 EC50 > 10000 nM T28893 CHA8V5 46890734 EC50 > 10000 nM T28893 CP7M3C 46890735 EC50 > 10000 nM T28893 CGYW61 46890736 EC50 > 10000 nM T28893 C5DTV6 46890737 EC50 > 10000 nM T28893 CPWD04 46890738 EC50 > 10000 nM T28893 CDT24N 46890774 EC50 > 10000 nM T28893 CQ0M8J 46890775 EC50 > 10000 nM T28893 CT82CV 46890776 EC50 > 10000 nM T28893 CV38XU 46890777 EC50 > 10000 nM T28893 C18WAP 46890778 EC50 > 10000 nM T28893 CP1VD4 46890779 EC50 > 10000 nM T28893 CWLF02 46890786 EC50 > 10000 nM T28893 CMA10I 46890787 EC50 > 10000 nM T28893 CN9B5A 46890788 EC50 > 10000 nM T28893 CZC91A 46890789 EC50 > 10000 nM T28893 C5GVQ6 46890790 EC50 > 10000 nM T28893 C5DPO2 46890846 EC50 = 3162.28 nM T28893 C0O4JF 46890847 EC50 = 7943.28 nM T28893 CAC73V 46890848 EC50 > 10000 nM T28893 CH6A4O 46890849 EC50 > 10000 nM T28893 CXK64W 46890850 EC50 > 10000 nM T28893 CF59KO 46890851 EC50 > 10000 nM T28893 C5NL8A 46890861 EC50 > 10000 nM T28893 C8O4HI 46890862 EC50 > 10000 nM T28893 C26EBN 46890863 EC50 > 10000 nM T28893 CBDL94 46890864 EC50 > 10000 nM T28893 CQ1P3Y 46890865 EC50 > 10000 nM T28893 CBT1C5 46890866 EC50 > 10000 nM T28893 C30KJT 46890906 EC50 = 1 nM T28893 CMCH59 46890907 EC50 = 1000 nM T28893 C81EPN 46890908 EC50 > 10000 nM T28893 CRH49B 46890909 EC50 > 10000 nM T28893 CJ59VT 46890910 EC50 > 10000 nM T28893 C7UV8K 46890911 EC50 = 398.11 nM T28893 C84EUG 46890919 EC50 > 10000 nM T28893 C7TMF3 46890920 EC50 > 10000 nM T28893 CI4KG6 46890921 EC50 > 10000 nM T28893 C6JF9I 46890922 EC50 > 10000 nM T28893 COI06F 46890923 EC50 > 10000 nM T28893 CU71IL 46890924 EC50 > 10000 nM T28893 CJ57WZ 46890960 EC50 = 501.19 nM T28893 C4GN3P 46890961 EC50 > 10000 nM T28893 CD1MS4 46890962 EC50 = 158.49 nM T28893 C8QZ2Y 46890963 EC50 = 50.12 nM T28893 CG2BK1 46890964 EC50 > 10000 nM T28893 CQO2W5 46890965 EC50 > 10000 nM T28893 CUA03J 46890972 EC50 = 1000 nM T28893 CYSD56 46890973 EC50 > 10000 nM T28893 C3FE1N 46890974 EC50 > 10000 nM T28893 C4VCD5 46890975 EC50 = 25.12 nM T28893 C39BYD 46890976 EC50 = 50.12 nM T28893 CW70YU 46890977 EC50 = 12.59 nM T28893 C72QOI 46891019 EC50 = 1584.89 nM T28893 C0KDX8 46891020 EC50 = 63.1 nM T28893 CJ10MI 46891021 EC50 = 501.19 nM T28893 CM01DZ 46891022 EC50 = 31.62 nM T28893 C3SQR9 46891023 EC50 > 10000 nM T28893 C17FOL 46891027 EC50 > 10000 nM T28893 CJ1O2Y 46891028 EC50 > 10000 nM T28893 CZUV58 46891029 EC50 = 1584.89 nM T28893 C7WJE3 46891030 EC50 = 39.81 nM T28893 C7KE4S 46891031 EC50 = 158.49 nM T28893 CO3XW8 46891074 EC50 > 10000 nM T28893 CZ1EO8 46891075 EC50 = 19.95 nM T28893 CJ74AZ 46891076 EC50 = 3.162 nM T28893 CSO96M 46891077 EC50 = 158.49 nM T28893 CMCD56 46891083 EC50 > 10000 nM T28893 CRH4V3 46891084 EC50 > 10000 nM T28893 CC10ZM 46891085 EC50 > 10000 nM T28893 CD5T4F 46891086 EC50 > 10000 nM T28893 C37BAT 46891087 EC50 > 10000 nM T28893 C8VCY5 46891140 EC50 = 25.12 nM T28893 CI9J3P 46891141 EC50 = 39.81 nM T28893 C6P5JG 46891142 EC50 = 158.49 nM T28893 C6I8NE 46891143 EC50 = 158.49 nM T28893 CW03QZ 46891144 EC50 = 63.1 nM T28893 C48SJN 46891149 EC50 > 10000 nM T28893 C1M9LF 46891150 EC50 > 10000 nM T28893 CR0T8P 46891151 EC50 > 10000 nM T28893 C1DVZ9 46891152 EC50 > 10000 nM T28893 C31CNM 46891153 EC50 > 10000 nM T28893 CTSZ49 46891179 EC50 = 10 nM T28893 CVZ07F 46891186 EC50 > 10000 nM T28893 COT8S4 46891375 EC50 = 251.19 nM T28893 CHC91G 46891376 EC50 = 251.19 nM T28893 CT4P1I 46891377 EC50 = 794.33 nM T28893 CWIH30 46891378 EC50 > 10000 nM T28893 CDR84O 46891379 EC50 > 10000 nM T28893 CHY81P 46891380 EC50 > 10000 nM T28893 CRBE14 46891431 EC50 > 10000 nM T28893 C5AHD3 46891432 EC50 > 10000 nM T28893 CBT8N5 46891433 EC50 > 10000 nM T28893 CFD7Q0 46891434 EC50 > 10000 nM T28893 CM7E8N 46891435 EC50 > 10000 nM T28893 C2Q0FT 46891436 EC50 > 10000 nM T28893 C4CLV8 46891484 EC50 > 10000 nM T28893 C5Y4HW 46891485 EC50 > 10000 nM T28893 CSCB34 46891486 EC50 > 10000 nM T28893 CA83LQ 46891487 EC50 > 10000 nM T28893 CW1YX7 46891488 EC50 = 63.1 nM T28893 CFQ1T7 46891489 EC50 = 86 nM T28893 C0H8WQ 46891544 EC50 > 10000 nM T28893 C5R4CZ 46891545 EC50 > 10000 nM T28893 C6AFP9 46891546 EC50 > 10000 nM T28893 C9C8NP 46891547 EC50 > 10000 nM T28893 CBOK70 46891548 EC50 > 10000 nM T28893 COP26M 46891549 EC50 > 10000 nM T28893 C61RTO 46891592 EC50 = 5011.87 nM T28893 C7XMN1 46891593 EC50 > 10000 nM T28893 C2O5RG 46891594 EC50 = 50.12 nM T28893 CDQ7B4 46891595 EC50 = 15.85 nM T28893 C0U6LX 46891596 EC50 > 10000 nM T28893 CF9YQ8 46891597 EC50 = 100 nM T28893 CB1Z5A 46905390 IC50 = 21.1 nM T28893 C2T8BK 46929965 EC50 = 150 nM T28893 CS73AB 46929966 EC50 = 49 nM T28893 C3DK2V 46929967 EC50 = 51 nM T28893 C61YXK 46929968 EC50 = 290 nM T28893 C5P1IE 46929969 EC50 = 560 nM T28893 CM3EZ8 46930073 EC50 = 120 nM T28893 C7HLQ9 46930074 EC50 = 1100 nM T28893 C1BPL4 46930170 EC50 = 910 nM T28893 CGA3R4 46930249 EC50 = 970 nM T28893 CV8E4X 46930250 EC50 = 27 nM T28893 CH5GY4 46930252 EC50 = 160 nM T28893 C90KRD 46930253 EC50 = 350 nM T28893 CD4G6O 46930341 EC50 = 9 nM T28893 CQWE65 46930342 EC50 = 20 nM T28893 CK8N6L 46930343 EC50 = 10 nM T28893 C67XQI 46945663 EC50 > 30000 nM T28893 C7IAW9 49663949 IC50 < 1500 nM T28893 CD39WZ 49665121 IC50 = 2800 nM T28893 C2LZJ0 49783209 Ki > 10000 nM T28893 C57SMG 49783415 Ki > 10000 nM T28893 C0TG6I 49783419 Ki > 10000 nM T28893 CC4KA6 49796398 IC50 = 35600 nM T28893 CKV07B 49796399 IC50 = 81 nM T28893 CRO0Y9 49796400 IC50 = 57 nM T28893 CJT93X 49796401 IC50 = 287 nM T28893 CM26YZ 49796402 IC50 = 79 nM T28893 C7V8HR 49796403 IC50 = 82 nM T28893 C8K3OZ 49796404 IC50 = 11500 nM T28893 C6PCF3 49796405 IC50 = 1217 nM T28893 C6MZS7 49796406 IC50 = 17700 nM T28893 CGD65N 49796407 IC50 = 1860 nM T28893 CF2W3N 49796408 IC50 = 1641 nM T28893 CCZ68J 49796409 IC50 = 131 nM T28893 CP6KL7 49796410 IC50 = 23500 nM T28893 CD4N3Q 49796411 IC50 = 44 nM T28893 CV0WH1 49796412 IC50 = 132700 nM T28893 C20SCO 49797320 Ki = 6141 nM T28893 C29QSB 49797322 Ki = 819 nM T28893 CT4QU7 49797325 Ki = 4550 nM T28893 CGB63L 49799920 EC50 = 159 nM T28893 CPI6N0 49853777 IC50 > 100000 nM T28893 C94GDK 49853778 IC50 > 100000 nM T28893 CHV3U8 49853881 IC50 > 100000 nM T28893 CTBY97 49853883 IC50 = 56000 nM T28893 CQP63D 49853884 IC50 = 50000 nM T28893 CY8M9A 49853885 IC50 > 100000 nM T28893 CN0JU9 49853987 IC50 > 100000 nM T28893 C8DVX6 49855131 IC50 = 102000 nM T28893 C2RY0J 50878551 Ki > 10000 nM T28893 C1W6TV 50898777 Ki > 10000 nM T28893 CXMZ73 50898778 Ki > 10000 nM T28893 CE4KP1 51050257 Ki > 10000 nM T28893 CM47HJ 52176747 IC50 = 1300 nM T28893 C6KU3Z 53303986 EC50 = 110 nM T28893 CS1OI7 53382523 EC50 > 30000 nM T28893 CWR16G 53382542 EC50 = 970 nM T28893 C7YP3A 53385782 EC50 = 17 nM T28893 CPGC12 53385783 EC50 = 350 nM T28893 C8V6IT 53385831 EC50 = 1200 nM T28893 CPR76N 53385877 EC50 = 320 nM T28893 C6A7VE 53414666 Ki = 18000 nM T28893 C6D3OU 54580864 IC50 = 1.1 nM T28893 CM9KH3 54581928 IC50 = 33.3 nM T28893 C1ZMV9 54582844 IC50 = 2.4 nM T28893 CMRC75 54583839 IC50 = 26.7 nM T28893 CZ82MJ 54583840 IC50 = 1 nM T28893 C01VQF 54584800 IC50 = 8.8 nM T28893 CHP9F8 54585742 IC50 = 319.4 nM T28893 CO5H6T 54585743 IC50 = 1.5 nM T28893 CB5IF2 54586723 IC50 = 428 nM T28893 CKTW24 54586742 IC50 = 9.2 nM T28893 CWXP12 54586744 IC50 = 3 nM T28893 C8WHT5 56593934 Ki = 10000 nM T28893 CB0P9N 56944383 Ki > 1000 nM T28893 C1TC7Q 56963799 Ki = 931 nM T28893 C3WC7Z 56965018 Ki = 4.571 nM T28893 CWT0H6 57105688 IC50 > 10000 nM T28893 CUP4Y0 57326139 Ki = 15488.17 nM T28893 C1G9XY 57326141 Ki > 100000 nM T28893 CG3YS9 57326143 Ki = 6760.83 nM T28893 CCYU25 57326145 Ki = 26302.68 nM T28893 CS86GL 57326232 Ki = 16.22 nM T28893 C3AF0Z 57326234 Ki = 0.5012 nM T28893 CLSW35 57326236 Ki = 3801.89 nM T28893 CL3R5D 57326238 Ki = 15848.93 nM T28893 C4G1LB 57326325 Ki = 35.48 nM T28893 C6CB9J 57326326 Ki = 1.259 nM T28893 C5OJP0 57391102 EC50 = 890 nM T28893 CX6AV8 57391280 IC50 > 10000 nM T28893 C8BO4V 57391281 IC50 > 10000 nM T28893 CJO67A 57391282 IC50 = 2100 nM T28893 C2AR3V 57391609 IC50 > 10000 nM T28893 CKPB03 57391802 IC50 > 10000 nM T28893 C8SW9E 57391803 IC50 > 10000 nM T28893 C5UWC6 57391804 IC50 > 10000 nM T28893 C78QEY 57391805 IC50 > 10000 nM T28893 CYAQ83 57391806 IC50 > 10000 nM T28893 COL58X 57391831 IC50 > 10000 nM T28893 CV8IK1 57393064 IC50 = 4800 nM T28893 C17GMJ 57393065 IC50 = 400 nM T28893 CKS3X9 57393534 IC50 > 10000 nM T28893 CM2EH0 57393535 IC50 > 10000 nM T28893 CNP60T 57393564 IC50 > 10000 nM T28893 CVO5M3 57393573 Ki > 10000 nM T28893 C5USX7 57395248 IC50 > 10000 nM T28893 CJ80BU 57395249 IC50 > 10000 nM T28893 C27MRL 57395273 IC50 > 10000 nM T28893 CX5MG4 57395274 IC50 > 10000 nM T28893 C40WGY 57395275 IC50 > 10000 nM T28893 C01VOH 57395286 Ki > 10000 nM T28893 CB48LK 57396543 IC50 > 10000 nM T28893 C42MVA 57396544 IC50 > 10000 nM T28893 C6HBG0 57396813 IC50 = 2200 nM T28893 C0P8KM 57397016 IC50 > 10000 nM T28893 CE85SV 57397017 IC50 > 10000 nM T28893 C0J9MO 57397044 IC50 > 10000 nM T28893 CCZ61A 57397045 IC50 > 10000 nM T28893 CZJ1P7 57397046 IC50 > 10000 nM T28893 CYC1Q5 57397055 Ki > 10000 nM T28893 C25FTZ 57397056 Ki = 340 nM T28893 CUP9S3 57398240 IC50 > 10000 nM T28893 CSU2O9 57398779 IC50 > 10000 nM T28893 C75ZGA 57399888 IC50 > 10000 nM T28893 CHKD69 57399987 IC50 > 10000 nM T28893 C5FDN6 57399988 IC50 > 10000 nM T28893 CW8TD0 57399989 IC50 > 10000 nM T28893 CUJ0A2 57399990 IC50 > 10000 nM T28893 CDQ57A 57400458 IC50 > 10000 nM T28893 CED9C4 57400459 IC50 > 10000 nM T28893 CSEK63 57400487 IC50 > 10000 nM T28893 CH6YT2 57400488 IC50 > 10000 nM T28893 CX0N7O 57400489 IC50 > 10000 nM T28893 CR0BU6 57400501 Ki = 430 nM T28893 CE82XL 57400502 Ki > 10000 nM T28893 CWZ50O 57400503 Ki = 930 nM T28893 C5MG6Q 57400504 Ki = 230 nM T28893 CJBU02 57400505 Ki > 10000 nM T28893 CDV7J0 57401665 IC50 > 10000 nM T28893 C0ESJ2 57401674 IC50 > 10000 nM T28893 CL52KE 57401786 IC50 > 10000 nM T28893 CV2ME6 57402260 IC50 > 10000 nM T28893 CQ1A8P 57402261 IC50 > 10000 nM T28893 CW94QA 57402262 IC50 > 10000 nM T28893 CMJA69 57402263 IC50 > 10000 nM T28893 CV2CF5 57402294 IC50 > 10000 nM T28893 CXT2L1 57402315 Ki > 10000 nM T28893 CUK9W4 57403507 IC50 > 10000 nM T28893 CX31VN 57403989 IC50 > 10000 nM T28893 C4E7UI 57404016 IC50 > 10000 nM T28893 C5FHR8 57404017 IC50 > 10000 nM T28893 C49JDH 57404030 Ki = 480 nM T28893 CQ5BG6 57525860 EC50 > 30000 nM T28893 C9TMZ3 57558000 Ki > 100000 nM T28893 CR7KU6 57845728 IC50 = 225 nM T28893 CA14SG 58653718 Ki > 100000 nM T28893 C2XDJ0 58975257 IC50 = 3829 nM T28893 CRV9X7 59654579 EC50 = 20.9 nM T28893 CDX98T 59691557 IC50 = 89 nM T28893 CUAY97 59691584 IC50 = 625 nM T28893 CDB34N 59691661 IC50 = 511 nM T28893 CV8U3A 59691704 IC50 = 446 nM T28893 C1MVB2 59835725 IC50 > 10000 nM T28893 CZ6EF7 59835728 IC50 = 2210 nM T28893 CMG1L8 59835758 IC50 = 2890 nM T28893 CG7JS4 59835780 IC50 = 285 nM T28893 C42PAO 59835879 IC50 = 665 nM T28893 C8HYR7 60130337 IC50 = 877 nM T28893 C35LSR 62705150 IC50 > 10000 nM T28893 C4VLW5 62705151 IC50 = 1800 nM T28893 C4R3SD 62705152 IC50 = 1700 nM T28893 CWUB45 62705153 IC50 = 2300 nM T28893 C5MN4X 62705154 IC50 = 1200 nM T28893 CR9E1J 62705155 IC50 = 2500 nM T28893 C02TAQ 62705172 EC50 = 12 nM T28893 CWL9J4 62705175 EC50 = 20 nM T28893 CQ5LS1 62705176 EC50 = 73 nM T28893 CNI52F 62705311 IC50 = 2290.87 nM T28893 CIG14S 62705312 IC50 > 10000 nM T28893 CH1S5G 62705313 IC50 = 831.76 nM T28893 CB15RK 62705314 IC50 = 830 nM T28893 C5HY3C 62705315 IC50 = 370 nM T28893 CLB26J 62705316 IC50 = 501.19 nM T28893 C59QUB 62705330 EC50 = 1700 nM T28893 CANL67 62705331 EC50 = 1200 nM T28893 C1SNE7 62705334 EC50 = 68 nM T28893 C63DKE 62705483 IC50 = 309.03 nM T28893 CAQZ57 62705484 IC50 = 1300 nM T28893 CHR98D 62705485 IC50 > 10000 nM T28893 CXEV16 62705486 IC50 > 10000 nM T28893 C15NVF 62705487 IC50 = 130 nM T28893 CAZ9B3 62705488 IC50 = 110 nM T28893 CZHO61 62705505 EC50 = 300 nM T28893 CP9HO0 62705507 EC50 = 44 nM T28893 CSHR51 62705508 EC50 = 66 nM T28893 CVPW40 62705509 EC50 = 110 nM T28893 C0X5NC 62705656 IC50 = 740 nM T28893 CW04AO 62705657 IC50 = 1548.82 nM T28893 C6UFJ9 62705658 IC50 = 2137.96 nM T28893 CV4ML9 62705659 IC50 = 1500 nM T28893 C5YWU7 62705660 IC50 = 180 nM T28893 CZ2NM6 62705661 IC50 = 690 nM T28893 C5S3JZ 62705830 IC50 = 512.86 nM T28893 CYJ6L2 62705831 IC50 = 107.15 nM T28893 C9F4JW 62705832 IC50 = 229.09 nM T28893 C7DQM1 62705833 IC50 > 10000 nM T28893 CW6GM7 62705834 IC50 = 2700 nM T28893 CIVC45 62705835 IC50 = 2818.38 nM T28893 CU6I5V 62706007 IC50 = 2000 nM T28893 CEO7M9 62706008 IC50 = 1900 nM T28893 CJ0NM6 62706009 IC50 = 1500 nM T28893 C49GQU 62706010 IC50 = 3162.28 nM T28893 C6PZ0O 62706011 IC50 = 1479.11 nM T28893 CQ52MB 62706173 IC50 = 5495.41 nM T28893 CX6GN3 62706488 IC50 > 10000 nM T28893 CBJ1M0 62706661 IC50 > 10000 nM T28893 C29LVW 62706662 IC50 = 2089.3 nM T28893 C53PIW 62707584 IC50 = 2500 nM T28893 CUO18E 62707585 IC50 = 1698.24 nM T28893 C3BJ1Y 62707586 IC50 = 2800 nM T28893 C49NOY 62707587 IC50 = 4073.8 nM T28893 CG4S1C 62707588 IC50 > 10000 nM T28893 CM0Z3B 62707610 EC50 = 6.3 nM T28893 CA5FP7 66561966 Ki = 5541 nM T28893 C3XL7O 66561967 Ki = 7958 nM T28893 C9A8WH 66875589 Ki = 0.5012 nM T28893 CB06GE 67547652 IC50 = 30.1 nM T28893 CDH6V7 67547661 IC50 = 290.8 nM T28893 CE91TN 67547949 IC50 = 76 nM T28893 CMA5W7 67548135 IC50 = 2.1 nM T28893 C8OC2K 67548543 IC50 = 281.4 nM T28893 CD41JS 67548925 IC50 = 1 nM T28893 C8MU9E 67549179 IC50 = 9.8 nM T28893 C4F7RP 68153829 EC50 = 1.2 nM T28893 CTJ26Q 68176440 EC50 = 2430 nM T28893 CCB1T5 68764898 Ki = 341 nM T28893 CTW10U 69058945 Ki = 1.585 nM T28893 C6TI9M 69444105 IC50 = 48.3 nM T28893 CF8DC9 70681307 Ki = 12.59 nM T28893 C7GP9T 70681453 EC50 = 1500 nM T28893 CTA92E 70681454 EC50 = 2500 nM T28893 C6JA0U 70682148 IC50 = 430 nM T28893 CXT67P 70683405 Ki = 45.71 nM T28893 CP86BK 70683564 EC50 = 3200000 nM T28893 C81BFH 70683565 EC50 > 10000 nM T28893 CE14HL 70683567 EC50 = 5400 nM T28893 CLX46N 70683569 EC50 = 3600 nM T28893 CN98LU 70685504 Ki = 6.31 nM T28893 C78XSZ 70685586 EC50 > 10000 nM T28893 C7X0WZ 70685587 EC50 = 1000 nM T28893 CA2N4J 70685669 EC50 = 6200000 nM T28893 C3MQ8V 70685670 EC50 = 1200000 nM T28893 COXJ45 70685676 EC50 = 1200 nM T28893 CYFC38 70685678 EC50 = 1100 nM T28893 CT41UM 70687661 Ki = 22.39 nM T28893 C7YB2Q 70687733 EC50 = 2000 nM T28893 C8QKZ4 70687825 EC50 = 4100000 nM T28893 CUHJ63 70687828 EC50 = 2000 nM T28893 CB6F3H 70687830 EC50 = 830 nM T28893 C7VXU0 70689860 EC50 = 470000 nM T28893 CEDV63 70689861 EC50 > 10000 nM T28893 C14QVU 70689864 EC50 = 2200 nM T28893 CEJP14 70689865 EC50 = 1900 nM T28893 CDOX61 70691923 EC50 = 570 nM T28893 CDT65S 70691924 EC50 > 10000 nM T28893 C80CVF 70692018 EC50 = 2100 nM T28893 CQK56J 70692022 EC50 > 10000 nM T28893 C9WYU5 70692024 EC50 = 440 nM T28893 CLC75M 70692025 EC50 = 810 nM T28893 CC7OG3 70694061 EC50 > 10000 nM T28893 C8LRI5 70694062 EC50 = 2300 nM T28893 CC43QK 71151588 Ki > 1000 nM T28893 C8OGT4 71283628 IC50 = 5000 nM T28893 CJLS94 71449148 Ki = 113.1 nM T28893 CQU65H 71449758 IC50 = 2398.83 nM T28893 CT4A3X 71449759 IC50 = 44 nM T28893 C24PKA 71449760 IC50 = 263.03 nM T28893 C7F3OR 71449761 IC50 = 1995.26 nM T28893 C4M1WQ 71450615 IC50 = 584.3 nM T28893 C29VNS 71450616 IC50 = 13.1 nM T28893 CDN70A 71450617 IC50 > 3300 nM T28893 C8HR1L 71450662 IC50 = 734.4 nM T28893 C8MQ6E 71451569 IC50 = 880 nM T28893 CY3M8B 71451570 IC50 = 17.78 nM T28893 CPB38T 71451571 IC50 = 33 nM T28893 C7WE6K 71451572 IC50 > 10000 nM T28893 CCH35F 71451573 IC50 > 10000 nM T28893 CG7M2C 71451574 IC50 = 89.13 nM T28893 C4NDR3 71452382 Ki = 32 nM T28893 C54WNK 71452454 IC50 > 3300 nM T28893 CPO41L 71452455 IC50 = 2497.4 nM T28893 CYF3R2 71452456 IC50 > 3300 nM T28893 C5WK8L 71452756 Ki = 0.68 nM T28893 CK81FI 71452793 Ki = 69.5 nM T28893 C6TG2S 71453412 IC50 > 10000 nM T28893 C1QF6R 71453413 IC50 > 10000 nM T28893 CG4ZX5 71454212 IC50 = 476 nM T28893 CSJ16R 71454213 IC50 = 462.4 nM T28893 CRMC04 71454214 IC50 = 1352.3 nM T28893 CZS9G3 71454215 IC50 = 327.2 nM T28893 CR41KC 71454216 IC50 < 5 nM T28893 C5OBD0 71454217 IC50 > 3300 nM T28893 CX26PA 71454562 Ki = 136.3 nM T28893 CX35MW 71454563 Ki = 2.14 nM T28893 C9QO7L 71455109 IC50 > 10000 nM T28893 CUWC72 71455110 IC50 > 10000 nM T28893 CD8PU4 71455111 IC50 = 104.71 nM T28893 CVIY45 71455112 IC50 > 10000 nM T28893 C6G2HC 71455894 Ki = 4610 nM T28893 CJ9XD3 71455951 IC50 = 300 nM T28893 CQ98SO 71455965 IC50 = 893.5 nM T28893 CWZ6X0 71455966 IC50 = 141 nM T28893 C9N0HT 71455967 IC50 < 5 nM T28893 CS4TY5 71455968 IC50 = 1115.3 nM T28893 CLWS62 71455969 IC50 = 1429.2 nM T28893 CG0A4Q 71456920 IC50 > 10000 nM T28893 C6B9ZY 71456921 IC50 = 240 nM T28893 C58AXY 71456922 IC50 = 500 nM T28893 CH9R6C 71456923 IC50 = 2500 nM T28893 CP7JI0 71457691 Ki = 313 nM T28893 C82EXK 71457751 Ki = 1288.25 nM T28893 C3Z9KW 71457770 IC50 = 881.5 nM T28893 C63TRO 71457771 IC50 = 378.6 nM T28893 C56DYG 71457818 IC50 > 3300 nM T28893 C4ZFG8 71458775 IC50 = 138.04 nM T28893 C0UX4H 71458776 IC50 = 100 nM T28893 C0YGE5 71458777 IC50 > 10000 nM T28893 C39IXM 71458778 IC50 = 3801.89 nM T28893 CCN84G 71458779 IC50 > 10000 nM T28893 C60GRE 71458940 Ki = 8.8 nM T28893 C4LXW7 71458941 Ki > 1000 nM T28893 CQ64EL 71459689 IC50 = 756.5 nM T28893 CNKD53 71459690 IC50 < 5 nM T28893 C8Q2FH 71459691 IC50 = 948.4 nM T28893 CH9R6O 71459724 IC50 = 1895.6 nM T28893 COQ67L 71459971 Ki = 253.3 nM T28893 C4QF5D 71460585 IC50 = 38 nM T28893 C1ST7X 71460586 IC50 > 10000 nM T28893 C63UYS 71460588 EC50 = 28.18 nM T28893 C2OIW1 71461631 IC50 = 62.4 nM T28893 CG8F1C 71461681 Ki = 103.8 nM T28893 CH56CX 71462298 IC50 = 100 nM T28893 COXM62 71462299 IC50 = 370 nM T28893 C79ZHJ 71462300 IC50 = 575.44 nM T28893 C1TG4H 71462301 IC50 = 436.52 nM T28893 CB5V7J 71462302 IC50 > 10000 nM T28893 CKG3U2 71463133 IC50 > 3300 nM T28893 CCR43M 71463134 IC50 > 3300 nM T28893 C27RGM 71463135 IC50 = 417.9 nM T28893 C3AKB0 71463136 IC50 = 198.8 nM T28893 C8YC5D 71533547 EC50 = 2398.83 nM T28893 CO0H8Z 71540043 EC50 > 10000 nM T28893 CWZ03G 71540044 EC50 = 1258.93 nM T28893 C5JDL0 71540045 EC50 > 10000 nM T28893 CHN5R1 71540145 EC50 > 10000 nM T28893 CKS05M 71540146 EC50 > 10000 nM T28893 CXKS79 71540147 EC50 > 10000 nM T28893 CVI15E 71540148 EC50 = 3300 nM T28893 CBE2K0 71540267 EC50 = 3300 nM T28893 CEK10S 71540272 EC50 > 10000 nM T28893 C56QLF 71540383 EC50 > 10000 nM T28893 C0TMW5 71540384 EC50 = 3981.07 nM T28893 CH36JK 71540385 EC50 = 5600 nM T28893 CG95KT 71540387 EC50 > 10000 nM T28893 CG06WS 71540490 EC50 = 5128.61 nM T28893 CE2C3V 71540491 EC50 > 10000 nM T28893 C5DVX1 71540492 EC50 > 10000 nM T28893 C7GAZ9 71540493 EC50 = 3200 nM T28893 CT35WB 71540494 EC50 > 10000 nM T28893 C18TPU 71540495 EC50 > 10000 nM T28893 CF95BW 71555066 EC50 = 1900 nM T28893 C97BWU 71568897 EC50 > 10000 nM T28893 CIVG64 71568899 EC50 = 1995.26 nM T28893 CLV8F6 71568900 EC50 = 2600 nM T28893 CTLP08 71568901 EC50 > 10000 nM T28893 CV4G2P 71569052 EC50 = 4073.8 nM T28893 CN5X6F 71570486 EC50 > 10000 nM T28893 C3QF8V 71570487 EC50 > 10000 nM T28893 C9Q0DE 71570627 EC50 = 2884.03 nM T28893 CGX51Q 71570629 EC50 > 10000 nM T28893 CMS82B 71570630 EC50 = 3800 nM T28893 CJ2Q7M 71570631 EC50 > 10000 nM T28893 CG4ZT6 71570772 EC50 > 10000 nM T28893 CIE2Z4 71570774 EC50 > 10000 nM T28893 C28SUY 71570775 EC50 = 1584.89 nM T28893 CV4J3Z 71570776 EC50 = 5128.61 nM T28893 C1PTJ3 71570777 EC50 = 7413.1 nM T28893 CC2P6G 71570918 EC50 > 10000 nM T28893 CF5VW0 71570919 EC50 = 3200 nM T28893 C4ZYI6 71570920 EC50 = 4073.8 nM T28893 CY76MQ 71570921 EC50 > 10000 nM T28893 CH0F8C 71571062 EC50 > 10000 nM T28893 C6JOV0 71571063 EC50 = 6300 nM T28893 CY01FS 71571064 EC50 = 5000 nM T28893 CZN1G5 71571209 EC50 = 2454.71 nM T28893 CK3G8O 71571210 EC50 = 3000 nM T28893 C68UAI 71574174 Ki = 27000 nM T28893 CK3T7C 71574175 Ki > 100000 nM T28893 CBZ78V 71574176 Ki > 100000 nM T28893 C61VXZ 71574177 Ki > 100000 nM T28893 C5OQ7W 71574178 Ki > 100000 nM T28893 CI0HU8 71574179 Ki > 100000 nM T28893 C6U4XJ 71574180 Ki > 100000 nM T28893 C0ZDF2 71574268 Ki > 100000 nM T28893 C0R3KB 71574269 Ki > 100000 nM T28893 CJ4WU1 71574271 Ki > 100000 nM T28893 C8ORK4 71574275 Ki = 6160 nM T28893 CCA49H 71574365 Ki = 210 nM T28893 CRT07Q 71574367 Ki > 100000 nM T28893 C0E9SQ 71575024 Ki = 1730 nM T28893 CJ3H1M 71575025 Ki = 470 nM T28893 CR04XZ 71575026 Ki = 3060 nM T28893 C3MJ7B 71575027 Ki = 3290 nM T28893 C8XEB3 71575028 Ki > 100000 nM T28893 C0XWU1 71575029 Ki = 200 nM T28893 C09DIB 71575117 Ki = 100 nM T28893 CM5OX8 71575118 Ki = 560 nM T28893 CAS1M2 71575119 Ki = 240 nM T28893 CL3A8V 71575120 Ki = 810 nM T28893 CQ21RK 71575121 Ki > 100000 nM T28893 CN82HY 71575122 Ki = 1390 nM T28893 CDAH09 71575123 Ki = 200 nM T28893 CZP59X 71575219 Ki = 60 nM T28893 CGR20T 71575220 Ki = 11700 nM T28893 C95ZSD 71575221 Ki > 100000 nM T28893 CTA7V5 71575222 Ki > 100000 nM T28893 CT03QG 71575223 Ki = 410 nM T28893 CYS85C 71575224 Ki = 370 nM T28893 C4I8TD 71575225 Ki = 140 nM T28893 CP3OI1 71575336 Ki > 100000 nM T28893 CQUT29 71575337 Ki = 20 nM T28893 CE4L0U 71575338 Ki > 100000 nM T28893 CJ5VK2 71575339 Ki > 100000 nM T28893 CY1Q9O 71575447 Ki = 290 nM T28893 CEX7R3 71575448 Ki > 100000 nM T28893 CD48AB 71575449 Ki > 100000 nM T28893 C0VAJ8 71575450 Ki = 5400 nM T28893 CD86FK 71575451 Ki > 100000 nM T28893 CVR1Q3 71575452 Ki = 920 nM T28893 CL3YP2 71575453 Ki = 340 nM T28893 CLX37P 71575548 Ki = 510 nM T28893 CHB4M1 71575549 Ki = 880 nM T28893 C3LE4R 71575550 Ki = 330 nM T28893 C93ZCM 71575551 Ki = 2700 nM T28893 CNS4V8 71575552 Ki = 25300 nM T28893 CM9SQ2 71575553 Ki = 24400 nM T28893 CMTB67 71575554 Ki > 100000 nM T28893 C1XV6F 71575649 Ki = 6190 nM T28893 CKI50H 71575650 Ki = 7900 nM T28893 CTSL25 71575651 Ki > 100000 nM T28893 C89MPL 71575652 Ki = 5270 nM T28893 COY38T 71575653 Ki = 2430 nM T28893 CK6F1D 71575654 Ki = 8350 nM T28893 CM8UN7 71598549 IC50 > 30000 nM T28893 CPZH08 71599959 EC50 = 1995.26 nM T28893 C1OE9J 71607097 IC50 > 30000 nM T28893 C0H5GZ 71656258 EC50 > 10000 nM T28893 CI0GU8 71660496 IC50 > 48500 nM T28893 C9I1TX 71717914 Ki > 100000 nM T28893 CO1R6X 71718834 EC50 = 1800 nM T28893 C6YQ4H 71719475 EC50 = 12 nM T28893 C3FQY2 71806339 IC50 > 10000 nM T28893 CHE5O6 72545089 Ki > 100000 nM T28893 CI6D4E 72545091 Ki > 100000 nM T28893 CKFW54 72545094 Ki > 100000 nM T28893 CWLO54 72545096 Ki > 100000 nM T28893 C5D4PA 72545098 Ki > 100000 nM T28893 CR39AG 72545326 Ki > 100000 nM T28893 C5HLF7 72545329 Ki > 100000 nM T28893 CWH6T3 72548703 IC50 = 18 nM T28893 C7W4RH 72734860 Ki > 1000 nM T28893 C6ZA8H 72945087 EC50 = 133 nM T28893 CC65OA 73213195 Ki > 10000 nM T28893 CW83DK 73213196 Ki > 10000 nM T28893 C6G3FB 73345317 Ki = 55.1 nM T28893 C46HUP 73345823 Ki = 10.7 nM T28893 C6J0TM 73346336 Ki > 10000 nM T28893 CP6H5M 73348351 Ki > 1000 nM T28893 CQ5D3T 73348823 Ki = 1040 nM T28893 C58SJG 73349591 Ki > 100000 nM T28893 CA6Z1P 73349592 Ki > 100000 nM T28893 CQU21G 73349926 Ki = 8.9 nM T28893 C9Z1FO 73350398 Ki = 519 nM T28893 CDS4F1 73350931 Ki = 5861 nM T28893 CA8L9Y 73351145 Ki > 100000 nM T28893 CFYS90 73351430 Ki = 8.8 nM T28893 CY53ZG 73354391 Ki = 45.4 nM T28893 C4F7VK 73355415 Ki = 7468 nM T28893 CX7ZV3 73356454 Ki = 5.75 nM T28893 C2K5DS 73672762 EC50 = 352 nM T28893 CHV3W1 73774630 EC50 > 30000 nM T28893 C2E7QW 75201901 IC50 = 4900 nM T28893 C8IDL3 75306277 Ki > 1000 nM T28893 CC4NP6 75356563 Ki = 4200 nM T28893 C50CMV 76309752 Ki = 7.81 nM T28893 C2NE1Q 76309753 IC50 = 86 nM T28893 CU5D8H 76309755 IC50 = 812.8 nM T28893 C42UQX 76309756 IC50 = 847.4 nM T28893 CO2N6P 76309757 IC50 = 84.5 nM T28893 C43NME 76313419 EC50 = 18 nM T28893 C7M4NP 76313420 EC50 = 3600 nM T28893 CZ80LO 76313453 IC50 = 420 nM T28893 CFP71X 76313455 IC50 = 611.8 nM T28893 CNI0G8 76313457 IC50 = 734.4 nM T28893 C1Y9WZ 76316965 Ki = 413 nM T28893 CQ2AF0 76316968 IC50 = 55.6 nM T28893 CD3GN5 76316970 IC50 = 161.3 nM T28893 CC57IB 76320662 EC50 > 10000 nM T28893 CJX71S 76320688 Ki = 17.8 nM T28893 CP7T1M 76320689 IC50 = 210.3 nM T28893 CZ6C0O 76320691 IC50 = 257.9 nM T28893 CL7U5W 76320693 IC50 = 1394 nM T28893 CHZ0P7 76320694 IC50 = 518.1 nM T28893 C5JNZ1 76324306 EC50 = 47 nM T28893 CU1J4Z 76324307 EC50 = 240 nM T28893 C8YW4N 76324331 Ki = 50 nM T28893 C94FIP 76324333 IC50 = 15.2 nM T28893 CN2S3T 76324335 IC50 = 1964.3 nM T28893 CA42PY 76324336 IC50 = 117.3 nM T28893 CFHZ75 76327871 EC50 = 1000 nM T28893 CP1U7E 76327897 Ki = 130 nM T28893 C8S1PB 76327898 Ki = 454 nM T28893 C9ATZ7 76327899 IC50 = 33.4 nM T28893 CQ94CR 76327901 IC50 = 1206.8 nM T28893 CUQ4W3 76327902 IC50 = 349.2 nM T28893 CJFI50 76327903 IC50 = 75.8 nM T28893 C6H9KX 76331523 EC50 = 170 nM T28893 C1WZ5N 76331540 Ki = 9.3 nM T28893 C47EDP 76331541 Ki = 154 nM T28893 C5N6LG 76331542 Ki = 18.6 nM T28893 CB46FR 76331543 IC50 = 125.5 nM T28893 C37DAL 76335135 EC50 = 170 nM T28893 C6N9SI 76335136 EC50 = 200 nM T28893 CZ2W7R 76335137 EC50 = 690 nM T28893 C4G6RW 76335160 Ki = 2110 nM T28893 CM54ZS 76335161 Ki = 438 nM T28893 CI2LH9 86298473 EC50 = 980 nM T28893 CX13CW 86298474 EC50 > 10000 nM T28893 C2BM9L 89768534 EC50 > 30000 nM T28893 CB4Y7R 89768546 EC50 > 30000 nM T28893 CYX9R8 89777050 EC50 > 10000 nM T28893 C5MR9K 89777151 EC50 > 30000 nM T28893 CPO7V2 90644379 EC50 = 316.23 nM T28893 CO2JA8 90644380 EC50 = 416.87 nM T28893 CB8I6J 90644381 EC50 = 1584.89 nM T28893 CTZ9G6 90644382 EC50 = 389.05 nM T28893 C4RUP2 101882890 Ki = 1.023 nM T28893 CH97BM 117680178 EC50 > 10000 nM T28893 C7DQW9 117937642 EC50 = 9.8 nM T28893 C3UVI2 117937644 EC50 = 28.5 nM T28893 CWL08D 117937652 EC50 = 30.3 nM T28893 CFL6Y2 117937665 EC50 = 478 nM T28893 CMG3A8 117937668 EC50 = 1800 nM T28893 C9TP0Z 117937675 EC50 = 25.3 nM T28893 C3H7NI 117973690 EC50 = 101 nM T28893 CG57HE 118110248 EC50 = 794.33 nM T28893 CGX21H 118110250 EC50 = 691.83 nM T28893 CWR6I1 118112300 IC50 > 30000 nM T28893 CEPL21 118123942 EC50 = 812.83 nM T28893 C6VXQ7 118123991 EC50 = 2238.72 nM T28893 CDZ2M0 118124039 EC50 = 2100 nM T28893 CE0FL7 118124048 EC50 = 707.95 nM T28893 C7F9OM 118124052 EC50 = 7079.46 nM T28893 CVTK73 118124055 EC50 = 6309.57 nM T28893 C9AWN0 118124117 EC50 = 250 nM T28893 C83UVP 118124136 EC50 < 10000 nM T28893 C7KYE9 118124140 EC50 = 1600 nM T28893 CMS06Z 118124164 EC50 = 5888.44 nM T28893 C64COX 118124169 EC50 = 2137.96 nM T28893 C4YEG3 118663155 Ki = 19 nM T28893 CC3YS5 118706050 Ki > 100000 nM T28893 C6DXV9 118706052 Ki > 100000 nM T28893 CL4EO9 118706054 Ki > 100000 nM T28893 CR0C4V 118718321 IC50 = 24.5 nM T28893 C4JY5S 118719502 IC50 > 30000 nM T28893 CI8CR0 118719920 Ki = 77.62 nM T28893 CV1WX5 118719921 Ki = 6.761 nM T28893 CIAG59 118719922 Ki = 0.912 nM T28893 CC5Q8Y 118719923 Ki = 10.96 nM T28893 CC8R6U 118719924 Ki = 44.67 nM T28893 CT8KO4 118719925 Ki = 2511.89 nM T28893 C16DHZ 118719926 EC50 = 112.2 nM T28893 CLA06I 118719927 EC50 = 69.18 nM T28893 CF20SR 118719928 Ki = 281.84 nM T28893 C6N7HV 118719929 Ki = 123.03 nM T28893 C64BIA 118719930 Ki = 186.21 nM T28893 CG4ZV5 118719931 Ki = 29.51 nM T28893 C05OBV 118723724 Ki > 100000 nM T28893 C5Z7FX 118724589 EC50 = 310 nM T28893 C2A4CM 118724592 EC50 > 10000 nM T28893 C3JSQ9 118724593 EC50 = 6309.57 nM T28893 CVWG17 118724594 EC50 > 10000 nM T28893 CBL9P1 118724596 EC50 = 656 nM T28893 C9LN6F 118724597 EC50 = 1412.54 nM T28893 C4ND5X 118724598 EC50 = 2020 nM T28893 CL0K6O 118724602 EC50 = 3790 nM T28893 C9YQT0 118724603 EC50 = 3630.78 nM T28893 C93DGV 118724604 EC50 = 1548.82 nM T28893 CKSJ43 118724605 EC50 = 812.83 nM T28893 CJ56GA 118724607 EC50 = 1940 nM T28893 C3XTQ0 118724608 EC50 = 1148.15 nM T28893 C7GEY3 118724611 EC50 = 0.6 nM T28893 CA17BK 118724612 EC50 = 10 nM T28893 C0Z5LI 118724613 EC50 > 30000 nM T28893 C4ONV3 118724614 EC50 > 10 nM T28893 C37MUF 118728610 IC50 = 6.1 nM T28893 C96QNO 118728611 IC50 = 176.7 nM T28893 CJU70M 118729452 EC50 = 5680 nM T28893 CG42YH 118729453 EC50 = 7540 nM T28893 C3TE5Z 118729455 EC50 = 17320 nM T28893 CCA76D 118729456 EC50 = 780 nM T28893 C76TDM 118732888 EC50 = 57.54 nM T28893 C5AJ7G 118732890 EC50 = 63.1 nM T28893 CTR19D 118732892 EC50 = 32.36 nM T28893 CH05JN 118732894 EC50 = 177.83 nM T28893 CYTK57 118732896 EC50 = 15.49 nM T28893 CV8XN9 118732898 EC50 = 302 nM T28893 CUBP10 118732900 EC50 = 58.88 nM T28893 C2KVL1 118732903 EC50 = 60.26 nM T28893 COS3K9 121304408 Ki = 457.09 nM T28893 C4RD9Y 121304424 Ki = 138.04 nM T28893 C1PKR0 121304441 Ki = 263.03 nM T28893 CC3MP6 121304452 Ki = 676.08 nM T28893 CW68KD 121304458 Ki = 741.31 nM T28893 CVA9F4 121304464 Ki = 169.82 nM T28893 COB2X5 121304477 Ki = 1659.59 nM T28893 CW51NQ 121304485 Ki = 309.03 nM T28893 C7NLV2 121304500 Ki = 251.19 nM T28893 CQ2UM4 121304538 Ki = 223.87 nM T28893 CN05ZQ 121304574 Ki = 302 nM T28893 CU0M7B 121304590 Ki = 478.63 nM T28893 CX5MO3 121304598 Ki = 173.78 nM T28893 C12GJP 121304609 Ki = 389.05 nM T28893 C31AEQ 121304649 Ki = 323.59 nM T28893 C2VTK5 121304654 Ki = 512.86 nM T28893 C5HQ4S 121304867 Ki = 562.34 nM T28893 CTJO50 122184561 IC50 = 8620 nM T28893 CZ1MA3 122184562 IC50 > 10000 nM T28893 CH37IW 122184563 IC50 = 2520 nM T28893 C5JTD9 122184564 IC50 > 10000 nM T28893 CJR48E 122184670 IC50 = 419 nM T28893 C7YA0Q 122184671 IC50 = 310 nM T28893 C6RP0N 122184672 IC50 = 3737 nM T28893 CLP36J 122184673 IC50 = 1920 nM T28893 C5Y0KX 122184691 IC50 = 1860 nM T28893 C18ZKO 122184692 IC50 > 10000 nM T28893 C0XJK1 122184693 IC50 > 10000 nM T28893 C97APV 122184694 IC50 > 10000 nM T28893 CLK94O 122184695 IC50 > 10000 nM T28893 CWSF63 122184696 IC50 > 10000 nM T28893 CW8L5K 122184697 IC50 > 10000 nM T28893 CI4SF6 122184698 IC50 = 5470 nM T28893 CDHE98 122184699 IC50 = 1650 nM T28893 CIU9W5 122184700 IC50 > 10000 nM T28893 CU2PG6 122184701 IC50 > 10000 nM T28893 CKG74I 122184702 IC50 = 2110 nM T28893 CZ0I1K 122184703 IC50 > 10000 nM T28893 C65COE 122184704 IC50 = 4470 nM T28893 CHS9N7 122184705 IC50 > 10000 nM T28893 CWM9Q7 122184706 IC50 > 10000 nM T28893 CD4ZG8 122186857 EC50 = 47.9 nM T28893 CR21ZV 122186858 EC50 = 71.5 nM T28893 CTV19U 122186859 EC50 = 11.1 nM T28893 CU48OE 122186860 EC50 = 34.8 nM T28893 CT3N9L 122186861 EC50 = 15.5 nM T28893 CL2T8A 122186862 EC50 = 9.1 nM T28893 C5X8MN 122186880 Ki > 10000 nM T28893 C3EZ7O 122189494 EC50 = 166 nM T28893 CKP85M 122189495 EC50 = 49.5 nM T28893 C2H3QF 122189496 EC50 = 36 nM T28893 C9HG5K 122189499 EC50 = 80 nM T28893 CAJ45R 122190994 EC50 = 51 nM T28893 C81TXF 122190995 EC50 = 118 nM T28893 CA3I7S 122190997 EC50 = 105 nM T28893 C15FXV 122190998 EC50 = 198 nM T28893 CYR7Q0 122190999 EC50 = 572 nM T28893 CIU6W4 122191000 EC50 = 837 nM T28893 C7TL4G 122191001 EC50 = 48.4 nM T28893 CA02ZK 122191002 EC50 = 87 nM T28893 CQI8E1 122191003 EC50 = 183 nM T28893 C80JRU 122191004 EC50 = 426 nM T28893 CF8N0T 122191005 EC50 = 154 nM T28893 C9G0TM 122191006 EC50 = 80.9 nM T28893 CR93HM 122191007 EC50 = 392 nM T28893 CRF36I 122191008 EC50 = 31 nM T28893 CX90IL 122194369 Ki = 10800 nM T28893 CU0B9P 122194370 Ki = 1200 nM T28893 C79UOH 122194371 Ki > 30000 nM T28893 CMY91C 122194372 Ki > 10000 nM T28893 CCDI50 122194373 Ki = 3630 nM T28893 C3JI4Q 122194374 Ki = 670 nM T28893 CA6M5R 122194375 Ki > 10000 nM T28893 C7M1QH 122194376 Ki = 3440 nM T28893 C1JB0D 122194377 Ki = 5090 nM T28893 CD5NB9 122194378 Ki = 2910 nM T28893 C8O1QD 122194379 Ki > 10000 nM T28893 CFYZ56 122194380 Ki = 5400 nM T28893 CQX7P1 122195090 EC50 = 14 nM T28893 C85FVS 124203829 Ki = 40 nM T28893 C89UBK 124415421 EC50 = 103 nM T28893 CCIA04 126492033 EC50 = 3630.78 nM T28893 C40FSB 126492034 EC50 = 1621.81 nM T28893 CHDO47 126492036 EC50 = 2290.87 nM T28893 C2FG0C 126492039 EC50 = 1174.9 nM T28893 CIV7R0 126533969 Ki = 1023.29 nM T28893 CIAD86 126534204 Ki = 1737.8 nM T28893 C4R7XU 126534291 Ki = 630.96 nM T28893 CVBX50 126534373 Ki = 109.65 nM T28893 C0WUJ5 126534771 Ki = 1000 nM T28893 C9Q0VB 126535075 Ki = 380.19 nM T28893 CZ61LK 127034966 EC50 > 5011.87 nM T28893 CA0SN5 127034967 EC50 > 5011.87 nM T28893 CUDA68 127038316 EC50 = 89 nM T28893 C5BCU2 127038317 EC50 = 185 nM T28893 C9H7BX 127038318 EC50 = 273 nM T28893 C0PMJ5 127038319 EC50 = 371 nM T28893 C8BWI1 127038324 EC50 = 63 nM T28893 CY6T0Q 127038325 EC50 = 112 nM T28893 CJCO32 127038678 EC50 = 248 nM T28893 C9F1TI 127038679 EC50 = 258 nM T28893 C3KIW1 127038680 EC50 = 500 nM T28893 CGYP61 127039038 EC50 = 163 nM T28893 CHC24D 127039039 EC50 = 4500 nM T28893 CA26DY 127039040 EC50 = 215 nM T28893 C9U0VA 127039041 EC50 = 255 nM T28893 CA4G1T 127039042 EC50 = 211 nM T28893 C34BGK 127040715 Ki = 1000 nM T28893 CS78AZ 127041951 Ki = 3162.28 nM T28893 CU9C4S 127041952 Ki = 1000 nM T28893 CV3OF2 127042157 EC50 = 175 nM T28893 C0ARE7 127042161 EC50 = 9 nM T28893 CQW02E 127042162 EC50 = 65 nM T28893 CJ2O5A 127044078 EC50 > 10000 nM T28893 CN50QE 127049132 EC50 > 10000 nM T28893 CE30QT 127049133 EC50 > 10000 nM T28893 C3WIA6 129103318 Ki > 1000 nM T28893 CJ94GK 129316454 Ki = 16 nM T28893 C50GOC 130442480 Ki = 8500 nM T28893 CM04RF 130442572 Ki = 9000 nM T28893 C4OC0I 132060752 Ki = 2473 nM T28893 CAVB41 132584404 Ki > 10000 nM T28893 CR8HL3 134134147 Ki = 371.54 nM T28893 CBU81N 134149168 Ki > 10000 nM T28893 C0S2VH 134150637 Ki = 66.07 nM T28893 C6NYU2 134150754 Ki = 489.78 nM T28893 CSK09D 134817226 EC50 = 210 nM T28893 C1GY2T 135156251 EC50 > 10000 nM T28893 C4UX2M 135430667 Ki = 7585.78 nM T28893 C72UDE 135493554 IC50 = 38 nM T28893 C0FG5R 135508767 IC50 = 27 nM T28893 C0TY5Z 135514603 IC50 = 54 nM T28893 C7RM9J 135515198 IC50 = 35 nM T28893 CB6OV7 135525247 Ki = 3 nM T28893 C2KG3B 135686415 IC50 = 19 nM T28893 CJI79M 136219242 Ki = 0.594 nM T28893 C63FEC 137125241 IC50 > 30000 nM T28893 CIHJ46 137125256 IC50 = 6 nM T28893 CR5FI1 137632077 EC50 = 18 nM T28893 C1PU6F 137633057 EC50 = 68 nM T28893 CI5SL0 137633162 Ki = 63 nM T28893 CD91UT 137634680 Ki = 7100 nM T28893 COI42G 137635637 EC50 = 4786.3 nM T28893 C6QB9W 137635734 Ki = 2290.87 nM T28893 CX8O0V 137636308 Ki = 2691.53 nM T28893 CRH92D 137636829 Ki = 7300 nM T28893 CWT0D8 137637047 Ki = 6100 nM T28893 CK61NA 137637129 EC50 = 50 nM T28893 C7VUW4 137637944 IC50 = 250 nM T28893 CY8Q1V 137638270 IC50 = 288 nM T28893 CFDB34 137639384 Ki = 17000 nM T28893 C4YJ1T 137639541 Ki = 20000 nM T28893 CV5C9P 137639937 EC50 = 24 nM T28893 CVIA23 137640095 Ki = 4900 nM T28893 CZ4TA9 137640201 EC50 = 186.21 nM T28893 CX4A3N 137640511 Ki = 12022.64 nM T28893 C2POD8 137640878 Ki = 42000 nM T28893 C70UDY 137641384 EC50 = 27 nM T28893 C8ZDW1 137642318 Ki = 7800 nM T28893 CXN8S4 137642540 EC50 = 26 nM T28893 C4Q6ZM 137642607 Ki = 2884.03 nM T28893 CW4IJ1 137644950 Ki = 38000 nM T28893 C0KL6Q 137644962 Ki = 1479.11 nM T28893 CG8P6I 137645938 Ki = 489.78 nM T28893 CO58KT 137646451 Ki = 330 nM T28893 CE5T3L 137646576 EC50 = 23 nM T28893 CJIU91 137647528 Ki = 13000 nM T28893 C2XMK6 137647734 IC50 = 313 nM T28893 CB9PL0 137648038 Ki = 1000 nM T28893 C3LC9W 137648483 Ki = 2500 nM T28893 CBN1K6 137650836 Ki = 7.079 nM T28893 C6WS1K 137653145 Ki = 17000 nM T28893 CFZS94 137653227 Ki = 20000 nM T28893 CCO85R 137653250 EC50 = 7 nM T28893 CWF8R1 137653324 Ki = 4500 nM T28893 C8XJO5 137653498 Ki = 380 nM T28893 C61WAG 137654353 IC50 = 540 nM T28893 C7DV5W 137654365 EC50 = 45 nM T28893 CC7GE8 137654674 Ki = 20000 nM T28893 CG49QD 137654747 EC50 = 36 nM T28893 CWOV78 137655063 IC50 = 322 nM T28893 CUC54G 137655636 Ki = 263.03 nM T28893 CUKT36 137655796 EC50 = 537.03 nM T28893 CUZ2V9 137656894 Ki = 1800 nM T28893 CQ2H0S 137657830 Ki = 170 nM T28893 CWSA41 137658091 Ki = 2900 nM T28893 C6E0JP 137659594 Ki = 23 nM T28893 C4BAP3 137660708 Ki = 16000 nM T28893 C7NJH0 137661079 Ki = 14000 nM T28893 C68QKL 137661317 Ki = 1.514 nM T28893 CDA8V2 137661377 Ki = 2511.89 nM T28893 C41ZYJ 137701968 EC50 = 320 nM T28893 CT78SZ 139413966 EC50 = 354 nM T28893 CRET23 139413979 EC50 = 70 nM T28893 CXWJ63 139414008 EC50 = 80 nM T28893 CFWM67 139414014 EC50 = 559 nM T28893 CMRB25 139414015 EC50 = 187 nM T28893 CP3Z2V 139414027 EC50 = 317 nM T28893 C30RNW 139414034 EC50 = 1465 nM T28893 CP0N7V 139414036 EC50 = 1469 nM T28893 CF15NK 139414044 EC50 = 238 nM T28893 C6SVB0 139414055 EC50 = 1846 nM T28893 CSR60Q 139414066 EC50 = 521 nM T28893 CD4IB3 139414069 EC50 = 251 nM T28893 C69RBA 139414071 EC50 = 232 nM T28893 CXU2W0 139414075 EC50 = 414 nM T28893 CJ6ZF7 139414093 EC50 = 104 nM T28893 CU5V8K 139414110 EC50 = 71 nM T28893 C59QBV 139414122 EC50 = 172 nM T28893 CYH5T8 139414129 EC50 = 420 nM T28893 CN8RU6 139414132 EC50 = 311 nM T28893 C12HNV 139414144 EC50 = 552 nM T28893 C7GH0M 139414161 EC50 = 50 nM T28893 C69DRM 139424615 EC50 = 649 nM T28893 C38OTS 145960427 Ki = 120.23 nM T28893 C06LVP 145960466 Ki = 4.571 nM T28893 C3WX5P 145960540 EC50 = 309.03 nM T28893 CSV5D4 145960592 Ki = 41.69 nM T28893 CR38AO 145960736 EC50 = 660.69 nM T28893 CXM0L2 145960766 EC50 = 478.63 nM T28893 C4KH9G 145960827 Ki = 54.95 nM T28893 C7LJZ2 145960875 EC50 = 2187.76 nM T28893 CP05YK 145961106 EC50 = 281.84 nM T28893 CJI6G2 145961125 Ki = 380.19 nM T28893 CK7OJ5 145961126 Ki = 660.69 nM T28893 CMB9T2 145961132 EC50 = 7300 nM T28893 C0XL7S 145961152 Ki = 1698.24 nM T28893 C3WFT9 145961161 Ki = 8.913 nM T28893 C9GI8W 145961193 EC50 = 1900 nM T28893 C2NK8O 145961235 EC50 = 2238.72 nM T28893 CQCO42 145961400 EC50 = 140 nM T28893 CYBS18 145961455 EC50 = 1258.93 nM T28893 CJ50OV 145961495 Ki = 67.61 nM T28893 C2FJX4 145961841 EC50 = 2800 nM T28893 CAH97Y 145961981 Ki = 194.98 nM T28893 CH1AE6 145962050 Ki = 190.55 nM T28893 CEXA18 145962138 EC50 = 3800 nM T28893 C4Y3JX 145962181 EC50 = 177.83 nM T28893 CX4J1C 145962519 EC50 = 3090.3 nM T28893 CO90NV 145962688 EC50 = 676.08 nM T28893 CXH76J 145962939 EC50 = 1071.52 nM T28893 CG16NQ 145963288 Ki = 162.18 nM T28893 C50RQB 145963344 EC50 = 2630.27 nM T28893 CD81FM 145963674 EC50 = 1400 nM T28893 CXE5L9 145963718 EC50 = 186.21 nM T28893 C85ZOK 145963821 IC50 = 1590 nM T28893 CR5AW1 145963843 EC50 > 10000 nM T28893 CU3D8E 145963886 EC50 = 275 nM T28893 CIZ2D6 145964146 IC50 = 3710 nM T28893 CL8IM7 145964214 IC50 = 5350 nM T28893 C9L6YX 145964246 EC50 > 10000 nM T28893 C6F5IU 145964557 EC50 = 165 nM T28893 CQH2M7 145965109 EC50 > 10000 nM T28893 CKQ0S8 145965599 EC50 = 349 nM T28893 CTH08B 145966538 EC50 > 10000 nM T28893 CZ20XJ 145967112 IC50 = 7860 nM T28893 CCVM34 145967131 IC50 = 4010 nM T28893 CYO7Q1 145967158 EC50 > 10000 nM T28893 C4BE0I 145968533 EC50 = 338 nM T28893 C3SHC0 145968558 EC50 = 34 nM T28893 CYNU03 145968963 EC50 > 10000 nM T28893 CC7O1U 145968975 EC50 = 99 nM T28893 C5U2KQ 145969027 EC50 = 70 nM T28893 CKQ3L7 145969071 EC50 > 300 nM T28893 C5ZMY6 145969333 EC50 = 162 nM T28893 CK10HF 145969354 EC50 = 12 nM T28893 C1HQW4 145969550 EC50 > 1101 nM T28893 CC1LA8 145969659 EC50 = 16 nM T28893 C52YHM 145969714 EC50 = 40 nM T28893 CUR83G 145970228 EC50 > 72 nM T28893 C2NEP6 145970252 EC50 = 63 nM T28893 C7KXI8 145970395 EC50 = 29 nM T28893 C7IN6K 145970758 EC50 > 10000 nM T28893 CJO3Z4 145970842 EC50 = 184 nM T28893 CFK7L2 145970884 EC50 > 3000 nM T28893 CY7FE0 145970887 EC50 > 1000 nM T28893 CG45PH 145970895 EC50 = 511 nM T28893 CTZ67D 145971059 EC50 > 207 nM T28893 CW81DQ 145971391 EC50 = 289 nM T28893 CKP39X 145971650 IC50 = 1070 nM T28893 C0RV3Z 145972056 IC50 = 2140 nM T28893 CJLK07 145972365 EC50 > 10000 nM T28893 C10KGM 145972388 IC50 = 2480 nM T28893 CE9U6I 145973015 IC50 = 4230 nM T28893 CQI6Y5 145973659 EC50 > 10000 nM T28893 CX31JO 145973665 EC50 > 10000 nM T28893 CR01XP 145973666 IC50 = 455 nM T28893 C2YZI7 145974021 EC50 > 10000 nM T28893 CP3W4L 145974148 IC50 = 4110 nM T28893 C7WRK1 145974265 IC50 = 3270 nM T28893 C9KNC3 145974491 IC50 = 2780 nM T28893 CXS48G 145974962 IC50 = 11400 nM T28893 C26ZBO 145975126 IC50 = 1370 nM T28893 C01XYS 145975344 EC50 > 10000 nM T28893 CI9UR8 145975401 EC50 = 267 nM T28893 CN3ZP2 145976302 EC50 = 399 nM T28893 CR1ZP7 145976328 EC50 = 62 nM T28893 C2WF3C 145976347 EC50 > 10000 nM T28893 CU1NO6 145976650 IC50 = 1490 nM T28893 CEXP52 145976876 IC50 = 8610 nM T28893 C4HWG1 145976924 EC50 > 10000 nM T28893 CD6C9H 145977656 EC50 > 10000 nM T28893 C5F3SW 145977820 EC50 > 10000 nM T28893 CYW3U1 145978073 IC50 = 658 nM T28893 CUD60Z 145978446 IC50 = 1480 nM T28893 CQ6TB5 145978697 IC50 = 9450 nM T28893 CE07DW 145978744 IC50 = 2050 nM T28893 CCG2I1 145982741 EC50 = 210 nM T28893 C61XIQ 145982857 EC50 = 60 nM T28893 CAD96U 145983366 EC50 = 660 nM T28893 CWJR39 145984661 EC50 = 89.13 nM T28893 C6W2KL 145985065 EC50 = 180 nM T28893 CR84PC 145985917 EC50 = 120 nM T28893 CQS04L 145986351 EC50 = 177 nM T28893 C2GX7C 145987038 EC50 > 249 nM T28893 CVZ2D6 145987046 EC50 > 257 nM T28893 CC2G1V 146025727 Ki = 6600 nM T28893 C6P3SR 153287553 Ki > 10000 nM T28893 CV9G7Z 153287572 Ki > 10000 nM T28893 CO85KL 153287574 Ki > 10000 nM T28893 CJKG35 155510347 Ki = 4300 nM T28893 C8IXK6 155511112 Ki = 590 nM T28893 CY83UA 155511167 Ki = 170 nM T28893 CUNX78 155511780 IC50 = 63.1 nM T28893 C2BDK6 155513985 Ki = 19.95 nM T28893 C6JSC8 155515662 Ki = 190 nM T28893 CUM2N4 155515982 Ki = 25000 nM T28893 CJG12Y 155516095 Ki = 710 nM T28893 C53FKW 155516382 Ki = 58.88 nM T28893 CI24NW 155516845 Ki = 780 nM T28893 CF9J5H 155517738 IC50 = 169.82 nM T28893 C0JM8H 155518181 Ki = 60 nM T28893 C3G2SA 155519666 IC50 = 323.59 nM T28893 C0MT4Q 155519740 Ki = 1.585 nM T28893 CUSA24 155519891 Ki > 10000 nM T28893 C4B7VK 155520267 Ki = 120 nM T28893 CPVA65 155521382 Ki = 97.72 nM T28893 C9N3JA 155521639 Ki = 1460 nM T28893 C7HPL3 155521847 Ki = 370 nM T28893 CFVP27 155521893 Ki = 2.138 nM T28893 CL9ET5 155522354 Ki = 41.69 nM T28893 CL6O1R 155523647 Ki = 0.871 nM T28893 C38PTA 155523888 Ki = 114.82 nM T28893 C8AMH9 155524478 Ki = 430 nM T28893 C6PFY7 155524809 Ki = 630 nM T28893 C5P1YE 155525064 Ki = 302 nM T28893 CDQ89Y 155525097 Ki = 1.445 nM T28893 C7UN0B 155525134 IC50 = 128.82 nM T28893 C7EIK1 155525691 Ki = 280 nM T28893 CBK0Y7 155528269 Ki = 95.5 nM T28893 CPG08Y 155528419 Ki = 760 nM T28893 CRPY78 155529196 Ki = 40 nM T28893 CU04AC 155531960 IC50 = 1.072 nM T28893 CN64WG 155534326 IC50 = 32.36 nM T28893 C8XHB9 155534466 IC50 = 15.14 nM T28893 C7CU8J 155535606 Ki = 2.754 nM T28893 CK91NV 155535972 Ki = 70 nM T28893 CB79ZW 155536080 Ki > 10000 nM T28893 C7AO1D 155536122 IC50 = 2089.3 nM T28893 C2XN8P 155536739 Ki = 70 nM T28893 CV2NG9 155539712 Ki = 2.344 nM T28893 CY2L3J 155540315 Ki = 770 nM T28893 CK70MJ 155541812 Ki = 2 nM T28893 CS5YB1 155543344 Ki = 177.83 nM T28893 COV93Z 155543943 Ki = 2.951 nM T28893 C17JEA 155543947 IC50 = 2200 nM T28893 C2CB8H 155548585 Ki = 107.15 nM T28893 C1XIA4 155549890 Ki = 690 nM T28893 C9KBH7 155550435 Ki = 1.413 nM T28893 CRIJ70 155550631 Ki = 1.23 nM T28893 CR8XF7 155551306 Ki = 200 nM T28893 CW92JZ 155551421 Ki = 1870 nM T28893 COF49W 155551902 Ki = 85.11 nM T28893 CX8JA1 155552185 Ki = 15000 nM T28893 CXZQ46 155552922 Ki = 87.1 nM T28893 CE70NU 155553089 Ki = 350 nM T28893 CS1DK6 155554149 Ki = 30 nM T28893 C7TF1D 155554261 Ki = 154.88 nM T28893 C73DFN 155554567 Ki = 3.162 nM T28893 C1TDY8 155556289 Ki = 1.259 nM T28893 C2D3SP 155557118 Ki = 93.33 nM T28893 C75PXS 155559290 Ki = 1047.13 nM T28893 CEAD84 155559740 Ki = 30.2 nM T28893 CP2U8A 155560012 Ki = 32.36 nM T28893 CU3TF1 155560139 Ki = 22.91 nM T28893 CCO15D 155560304 Ki = 2.399 nM T28893 CMX98Q 155562285 Ki = 10 nM T28893 C7P2OG 155562295 Ki = 770 nM T28893 CE8J7I 155562520 IC50 = 13.8 nM T28893 CDYV69 155562882 Ki = 790 nM T28893 C8WE2F 155563061 Ki = 6980 nM T28893 C2G7UH 155565074 Ki = 300 nM T28893 CVLR58 155565285 Ki = 537.03 nM T28893 C9AF7I 155565770 Ki = 95 nM T28893 CDS7K2 155566289 Ki = 2.291 nM T28893 CY30EN 155567379 Ki = 2.291 nM T28893 C3N9VU 10251906 Ki > 500 nM T28893 C9RLJ3 3661 Ki = 0.44 nM T28893 CD6OK3 44455198 Ki = 4.6 nM T28893 D01JXM 46222048 Ki > 1000 nM T28893 D01UDC 9815331 Ki = 4.6 nM T28893 D02BOW 5926 Ki = 1949.84 nM T28893 D02EXX 3013846 Ki = 490 nM T28893 D02KZD 71598521 IC50 > 30000 nM T28893 D02MJE 10426487 EC50 = 15.7 nM T28893 D02UNX 24768606 IC50 = 690 nM T28893 D02VGM 23056 Ki = 0.051 nM T28893 D02ZPV 10125445 Ki = 19.95 nM T28893 D03DKZ 42633508 EC50 > 30000 nM T28893 D04TWX 9794475 Ki > 1000 nM T28893 D04XNH 44318851 Ki = 190 nM T28893 D05EML 21847 IC50 < 1 nM T28893 D05ZUX 44207909 EC50 = 61 nM T28893 D06BSD 44405301 Ki = 69.7 nM T28893 D06IUC 6508730 Ki = 34 nM T28893 D06VST 15685977 IC50 = 2800 nM T28893 D07GPQ 132947 Ki = 1.585 nM T28893 D09HXG 10463948 Ki = 53.5 nM T28893 D09PIN 3378093 Ki > 1000 nM T28893 D09RPR 16737207 Ki > 10000 nM T28893 D0A2KT 3014059 Ki = 1.1 nM T28893 D0AR0H 6508724 Ki = 44 nM T28893 D0C2DM 9893054 EC50 = 22.8 nM T28893 D0C9VH 19718 IC50 = 87880 nM T28893 D0C9ZE 10105296 Ki = 120 nM T28893 D0F5LH 4634 Ki = 1 nM T28893 D0FF6S 16038374 IC50 > 10000 nM T28893 D0FX4W 10104167 IC50 = 1.259 nM T28893 D0G4CG 4629 EC50 = 7400 nM T28893 D0H2UT 442021 Ki = 44668.36 nM T28893 D0H4BJ 9308 Ki = 56 nM T28893 D0H8XV 12963076 Ki = 2.4 nM T28893 D0HP1O 119357 Ki = 12.4 nM T28893 D0I9LU 2229 Ki = 1230.27 nM T28893 D0JV2S 3008304 EC50 = 6000 nM T28893 D0L1XR 4630 Ki = 1.122 nM T28893 D0L5MW 181743 Ki > 10000 nM T28893 D0M0BM 10399068 IC50 = 6090 nM T28893 D0M2LD 1476756 EC50 < 100 nM T28893 D0M5ZE 5311416 Ki = 1584.89 nM T28893 D0O0LU 264734 EC50 = 10 nM T28893 D0P0IX 16104 IC50 = 6 nM T28893 D0P1FJ 71128 Ki = 2.1 nM T28893 D0R8FS 19816 IC50 = 51800 nM T28893 D0T2RY 9948320 EC50 = 150 nM T28893 D0T6ID 10062394 IC50 = 0.002 nM T28893 D0TX8W 594590 Ki > 19952.62 nM T28893 D0W9RR 57339144 IC50 = 3500 nM T28893 D0WO3A 4141 Ki = 7943.28 nM T28893 D0X7HD 11184481 Ki = 14000 nM T28893 D0Y8UC 3929516 Ki = 11.6 nM T28893 D0Z5RQ 656392 IC50 = 505 nM T28893 D0Z6VT 71737672 EC50 = 5400 nM T04911 D09ZZW 503536 IC50 = 1500 nM T04911 C6IQV0 482174 IC50 = 5700 nM T04911 CY61LO 487910 IC50 = 1700 nM T04911 C6K5JV 487911 IC50 = 16000 nM T04911 C3J5VH 487912 IC50 = 1000 nM T04911 CZNK70 487918 IC50 = 330 nM T04911 CDN3F2 487919 IC50 = 1630 nM T04911 CT76XW 487920 IC50 = 2100 nM T04911 CVA82G 487921 IC50 = 460 nM T04911 CBR46W 487922 IC50 = 1400 nM T04911 CAJ64Q 490750 IC50 < 1000 nM T04911 CMO49H 491114 IC50 = 4300 nM T04911 COB17R 492544 IC50 > 50000 nM T04911 C68MZE 492548 IC50 > 100000 nM T04911 C4JO9E 492549 IC50 = 3280 nM T04911 C1JEY2 492550 IC50 = 300 nM T04911 CRML27 492552 IC50 = 380 nM T04911 C84QRW 493418 IC50 = 5700 nM T04911 CY1WF7 497453 IC50 = 3000 nM T04911 C43PXV 503499 IC50 = 2400 nM T04911 C2BSI5 503516 IC50 = 14000 nM T04911 CFRT87 503517 IC50 = 5400 nM T04911 C3JB0U 503520 IC50 = 13000 nM T04911 CA72XJ 503521 IC50 = 5200 nM T04911 CF14KO 503522 IC50 = 7400 nM T04911 CH18YP 503523 IC50 = 4600 nM T04911 CG6T1D 503524 IC50 = 4100 nM T04911 CLY7T8 503525 IC50 = 750 nM T04911 C37MIA 503526 IC50 = 1000 nM T04911 C8U2AD 503527 IC50 = 12000 nM T04911 CO6R4G 503528 IC50 = 2000 nM T04911 CHA5F8 503529 IC50 > 50000 nM T04911 C41DVG 503530 IC50 = 21000 nM T04911 C5XRJ6 503531 IC50 = 1200 nM T04911 CI1V6W 503532 IC50 > 50000 nM T04911 C84DXH 503533 IC50 = 1400 nM T04911 C7R3CM 503534 IC50 = 2000 nM T04911 CCMU16 503535 IC50 = 3000 nM T04911 C1E4IO 504181 IC50 = 2700 nM T04911 CEJ6U1 504182 IC50 = 1800 nM T04911 CZDS90 504183 IC50 = 1600 nM T04911 C04ONL 504184 IC50 = 2200 nM T04911 C65XPH 504185 IC50 = 11000 nM T04911 CRZN68 504186 IC50 = 42000 nM T04911 CK8CA2 504187 IC50 > 60000 nM T04911 C01MYV 504188 IC50 = 5800 nM T04911 C4C5WD 504189 IC50 = 4300 nM T04911 CIB52E 504190 IC50 = 230 nM T04911 CQ6L1G 504191 IC50 = 12000 nM T04911 C4CW5A 504192 IC50 > 60000 nM T04911 C09ACU 504193 IC50 > 60000 nM T04911 C7T0AD 504194 IC50 = 1300 nM T04911 C7VZY1 504195 IC50 > 60000 nM T04911 CU4EK0 504196 IC50 = 3600 nM T04911 COUS53 504197 IC50 = 5300 nM T04911 CTE3B4 504198 IC50 = 7700 nM T04911 CT81MP 504676 IC50 = 3500 nM T04911 C9FI5K 504680 IC50 = 10600 nM T04911 C8IFN4 504681 IC50 = 31000 nM T04911 CV6OY3 506523 IC50 = 1400 nM T04911 CQX7S4 506524 IC50 = 390 nM T04911 CXD73I 506525 IC50 = 1800 nM T04911 C6ANI5 506528 IC50 = 9000 nM T04911 CRU30I 507613 IC50 = 900 nM T04911 CI8SQ4 511361 IC50 > 50000 nM T04911 C02LPN 511362 IC50 = 30000 nM T04911 CJIW67 511363 IC50 = 13000 nM T04911 C3KG1M 511364 IC50 = 43000 nM T04911 CU85HK 511365 IC50 = 10700 nM T04911 C20EKN 511366 IC50 = 5900 nM T04911 C3FX8J 511367 IC50 = 31000 nM T04911 C4DEY1 511368 IC50 = 3700 nM T04911 CC2J9M 511369 IC50 = 5600 nM T04911 CIU5M2 511370 IC50 = 11000 nM T04911 C5CG4I 511371 IC50 = 5000 nM T04911 CTO87P 511372 IC50 = 2700 nM T04911 C5BJ6S 511373 IC50 = 26000 nM T04911 CDWB40 511374 IC50 = 15000 nM T04911 CDH29C 511375 IC50 = 31000 nM T04911 C8ZJD7 511376 IC50 = 31000 nM T04911 CJ56OH 513150 IC50 < 10000 nM T04911 C5BN4U 513891 IC50 = 12000 nM T04911 CVI54C 657065 IC50 = 1200 nM T04911 CUC54L 3008068 IC50 = 5000 nM T04911 CJ5NO6 3008069 IC50 = 34000 nM T04911 CQO9Y3 3008070 IC50 > 32000 nM T04911 CXM1K9 3008071 IC50 > 50000 nM T04911 CJ2NY3 3008418 IC50 = 20000 nM T04911 CIJ2T0 3008419 IC50 > 50000 nM T04911 CWD1X0 3008420 IC50 = 14000 nM T04911 C4K2JP 3008421 IC50 > 50000 nM T04911 CAN83S 3008422 IC50 = 13000 nM T04911 CMDQ27 4468931 IC50 = 1800 nM T04911 CK9WY1 5278824 IC50 = 100 nM T04911 C5MEQ4 5278825 IC50 = 110 nM T04911 C1F0AN 5278826 IC50 = 45 nM T04911 CV0O6S 5482516 IC50 = 15600 nM T04911 CEM30Z 5483089 IC50 = 8900 nM T04911 CJL21S 9853197 IC50 = 60 nM T04911 CJW4M9 9917616 IC50 = 11000 nM T04911 C39ZBC 10207572 IC50 = 30000 nM T04911 CGA86Z 10259200 IC50 = 12000 nM T04911 CJ46UK 10439772 IC50 = 420 nM T04911 COM8C5 21148125 IC50 = 16000 nM T04911 C1TW3V 22209806 IC50 > 50000 nM T04911 C8GVX3 22209808 IC50 > 50000 nM T04911 C6AS7E 22209811 IC50 = 3300 nM T04911 CLW13P 22209812 IC50 = 1700 nM T04911 C1TA6Z 22209813 IC50 = 440 nM T04911 CGUC83 22210989 IC50 = 58000 nM T04911 CV97ER 22210996 IC50 = 18000 nM T04911 C2BA1K 22211000 IC50 = 27000 nM T04911 C78AKX 22211010 IC50 > 100000 nM T04911 CL7M9B 22211011 IC50 = 32000 nM T04911 C1L8TE 22211012 IC50 = 18000 nM T04911 C0NYS5 22211016 IC50 = 50000 nM T04911 C67QJW 22211018 IC50 > 100000 nM T04911 CV9S2O 22211019 IC50 = 13000 nM T04911 C4UB6Q 22211020 IC50 = 14000 nM T04911 CBUV46 22211021 IC50 = 62000 nM T04911 CS9B7N 22211022 IC50 > 100000 nM T04911 CK81WO 25078062 IC50 = 3400 nM T04911 CYDW71 44268661 IC50 > 60000 nM T04911 C6S3AT 44268682 IC50 > 60000 nM T04911 CDJ0X4 44308299 IC50 > 100000 nM T04911 CIO1C2 44308345 IC50 > 100000 nM T04911 CX14BI 44308422 IC50 > 100000 nM T04911 CE3PS8 44308752 IC50 = 34000 nM T04911 CK2P5O 44375061 IC50 > 50000 nM T04911 C4CVW1 44375110 IC50 > 50000 nM T04911 C72KUL 44375154 IC50 = 9400 nM T04911 C1SBO9 44375192 IC50 > 50000 nM T04911 C42GUE 44375229 IC50 = 5300 nM T04911 CX76FI 44388198 IC50 = 350 nM T04911 CVW6O4 44399745 IC50 = 79432.82 nM T04911 CDRP83 44399750 IC50 = 50118.72 nM T04911 CW6NY8 44399751 IC50 = 5011.87 nM T04911 CM5W8Q 44399752 IC50 = 6309.57 nM T04911 C34WSP 44399753 IC50 = 10000 nM T04911 CE0T1O 44399754 IC50 = 1995.26 nM T04911 CT86CR 44399784 IC50 = 25118.86 nM T04911 C6GWS9 44399837 IC50 = 31622.78 nM T04911 C4AI1T 44399861 IC50 = 100000 nM T04911 CTX79F 44399866 IC50 = 25118.86 nM T04911 CP4KB7 44399867 IC50 = 794.33 nM T04911 C0WRU5 44399868 IC50 = 15848.93 nM T04911 C8JP2A 44399889 IC50 = 50118.72 nM T04911 CO4H3V 44399938 IC50 = 10000 nM T04911 CYH7F9 44399975 IC50 = 6309.57 nM T04911 CZRF38 44399976 IC50 = 6309.57 nM T04911 CATH48 44399977 IC50 = 6309.57 nM T04911 CL9NS3 44399978 IC50 > 199526.23 nM T04911 C9YO4K 44399979 IC50 > 199526.23 nM T04911 CX8M3O 44400003 IC50 = 39810.72 nM T04911 C4X1OG 44400004 IC50 = 19952.62 nM T04911 C5EV1S 44400005 IC50 = 158489.32 nM T04911 CFRU27 44400006 IC50 = 199526.23 nM T04911 C7FO3T 44400007 IC50 = 251188.64 nM T04911 CA6P2U 44400008 IC50 = 100000 nM T04911 CQP47M 44400009 IC50 = 7943.28 nM T04911 CCRB97 44400010 IC50 = 3981.07 nM T04911 CT40SR 44400033 IC50 = 31622.78 nM T04911 CA96HO 44400076 IC50 > 1000000 nM T04911 CX7O2Z 44400112 IC50 > 199526.23 nM T04911 C6Z5NC 44400113 IC50 > 199526.23 nM T04911 C6PCE5 44400114 IC50 = 31622.78 nM T04911 C95CRD 44400115 IC50 = 19952.62 nM T04911 CW5G3Z 73347065 IC50 > 50000 nM T04911 C6TNQ8 135412361 IC50 = 800 nM T04911 C53AWL 135434400 IC50 = 100 nM T58772 D03DPZ 45375953 IC50 = 1 nM T58772 D03EZE 25167777 Ki = 0.18 nM T58772 D05EXN 58298316 IC50 = 30 nM T58772 D0O1IM 58298318 IC50 = 23 nM T58772 D0TU7B 58507717 IC50 = 205 nM T58772 D0VG0D 11977753 IC50 = 44 nM T58772 D0Z2UQ 25262792 IC50 = 200 nM T58772 D0K1VK 25262965 IC50 = 0.8 nM T58772 C2HY0V 5902454 IC50 = 1 nM T58772 CV9US5 16736978 IC50 = 660 nM T58772 C7QSC9 24905154 IC50 = 8 nM T58772 CH6Q7Y 24983749 IC50 = 2410 nM T58772 CK73NR 44219749 IC50 = 5 nM T58772 C1D4TK 46214389 IC50 = 53 nM T58772 C93ZNA 46215208 IC50 = 66 nM T58772 CGMS50 46215563 IC50 = 108 nM T58772 CO1D6B 46215565 IC50 = 230 nM T58772 CY8MP7 49867926 IC50 = 190 nM T58772 CRJ5W8 51358113 EC50 = 0.25 nM T58772 C9NS6B 52933960 IC50 = 85 nM T58772 CU3WG8 58298312 IC50 = 386 nM T58772 CONJ64 58298326 IC50 = 44 nM T58772 C0W7QE 58298327 IC50 = 10 nM T58772 C7GIQ1 58298333 IC50 = 650 nM T58772 CQ4HD1 59239114 IC50 = 9.1 nM T58772 CY3M0Z 59239164 IC50 = 7.8 nM T58772 CVG8B3 59239456 IC50 = 19 nM T58772 CI2SU0 59453028 IC50 = 6 nM T58772 CY8L4O 59453029 IC50 = 15 nM T58772 CTMA05 59453047 IC50 = 8 nM T58772 C8YDC3 59453057 IC50 = 240 nM T58772 CYN1L2 59453060 IC50 = 340 nM T58772 CV6A4J 59453078 IC50 = 46 nM T58772 CM2Q5J 59453081 IC50 = 4 nM T58772 CRFC53 59453089 IC50 = 20 nM T58772 C1RTQ6 59453093 IC50 = 240 nM T58772 C26QRA 59453105 IC50 = 54 nM T58772 C2BM8E 59453110 IC50 = 10 nM T58772 CXA9D8 59453133 IC50 = 200 nM T58772 C0X9FR 66699750 IC50 = 40 nM T58772 CIT38E 67179786 IC50 = 62 nM T58772 CA1WS0 67276196 IC50 = 35 nM T58772 C6E5BT 71243388 IC50 > 10000 nM T58772 C6T2UX 71243411 IC50 = 100 nM T58772 C82USW 71481184 IC50 = 100 nM T58772 C7V9SQ 71547699 IC50 = 14.5 nM T58772 COG0X5 71604742 IC50 = 8.2 nM T58772 CC5UR3 71604893 IC50 = 15 nM T58772 COZ4A6 71604894 IC50 = 7.4 nM T58772 C13FGZ 71604895 IC50 = 7.7 nM T58772 C4NA0Z 71604896 IC50 = 82 nM T58772 CNY35F 71604897 IC50 = 25 nM T58772 CN08ZO 71605054 IC50 = 15 nM T58772 CHK8Y6 71605056 IC50 = 8.2 nM T58772 C0HEN3 71605057 IC50 = 2.4 nM T58772 C5K9JV 71717638 IC50 = 1.3 nM T58772 C5S8DT 71717639 IC50 = 2 nM T58772 CJP83B 71719453 IC50 = 0.7 nM T58772 C86MQI 71720046 IC50 = 2.7 nM T58772 CLT60U 71720047 IC50 = 3.3 nM T58772 C28ZGR 73350474 IC50 = 1863 nM T58772 C7H4BN 73352721 IC50 > 10000 nM T58772 C72XAS 73353453 IC50 = 1000 nM T58772 C64QBH 117995822 IC50 = 164 nM T58772 C7KTW4 118000035 IC50 = 1790 nM T58772 CB0TU3 118000135 IC50 = 524 nM T58772 C0JC8U 118000139 IC50 = 751 nM T58772 C7E2DY 118000150 IC50 = 96 nM T58772 CKZ5N0 118000206 IC50 = 1857 nM T58772 C8M2ET 121334520 IC50 = 85.2 nM T58772 C3N2QP 122188110 IC50 = 78 nM T58772 C6O3MQ 136240948 IC50 = 1 nM T58772 C1QHU9 136259916 IC50 = 1 nM T58772 CJ2LR9 136259917 IC50 = 100 nM T58772 CDKR41 139030535 IC50 = 60 nM T58772 C1NQ0F 139207772 IC50 = 40 nM T58772 C3O5IA 139207773 IC50 = 8 nM T58772 CKLH15 139207774 IC50 = 4 nM T58772 C8FZE6 142608579 IC50 = 7 nM T58772 C1OVC9 155511557 IC50 = 55 nM T58772 C73TXJ 155513291 IC50 = 2655 nM T58772 CBK3C9 155515384 IC50 = 40 nM T58772 CBG61O 155518418 IC50 = 1239 nM T58772 CJMD34 155525139 IC50 = 240 nM T58772 C3I9UX 155526450 IC50 = 160 nM T58772 CPJ3R6 155526809 IC50 = 149 nM T58772 CJ3LP5 155528779 IC50 = 289 nM T58772 C9OVL5 155528904 IC50 = 60 nM T58772 CY9V8G 155530040 IC50 = 938 nM T58772 C68NQP 155536585 IC50 = 245 nM T58772 CE8TV9 155541005 IC50 = 45 nM T58772 CN5U9M 155541206 IC50 = 377 nM T58772 CV5L6B 155543139 IC50 = 420 nM T58772 C6JCV4 155548973 IC50 = 40 nM T58772 CJWV35 155549094 IC50 = 30 nM T58772 CE5DG7 155550972 IC50 = 432 nM T58772 CVO9N5 155551369 IC50 = 2520 nM T58772 C8L4MZ 155554924 IC50 = 826 nM T58772 CO4GE3 155557022 IC50 = 230 nM T58772 C61SQJ 155558592 IC50 = 43317 nM T58772 C6BAV3 155558720 IC50 = 136 nM T58772 CZCO50 155559160 IC50 = 2425 nM T58772 C7TP0F 155559332 IC50 = 354 nM T58772 C4GXV3 155562151 IC50 = 30 nM T58772 C6RV0H 155563416 IC50 = 7 nM T58772 CTEB79 155563891 IC50 = 132 nM T58772 C5SH4P 155565730 IC50 = 991 nM T58772 C3XMB6 155567232 IC50 = 35 nM T58772 CVR2J1 155569607 IC50 = 61 nM T58772 D0H0HR 49836027 IC50 = 2 nM T58772 D0H2CM 135565635 IC50 = 8 nM T58772 D0W8XH 9884685 IC50 = 20 nM T80165 D06XDJ 2782 IC50 = 11300 nM T80165 C6EM0S 1096735 IC50 = 500 nM T80165 C5E4RY 1096815 IC50 = 400 nM T80165 C5ADZ4 4519833 IC50 = 800 nM T80165 C1CBH5 12187315 IC50 = 1570 nM T80165 C3XJB2 17466271 IC50 > 30000 nM T80165 CY7O0L 53378752 IC50 = 7.9 nM T80165 C09LTC 56944680 IC50 = 160 nM T80165 CT29AF 71818278 IC50 = 800 nM T80165 CNQ38C 71818279 IC50 = 3160 nM T80165 C7APU4 71818280 IC50 = 630 nM T80165 C61GSX 71818281 IC50 = 160 nM T80165 C23DTZ 71818282 IC50 = 630 nM T80165 CQ20DY 71818427 IC50 = 15800 nM T80165 C5GI1E 71818428 IC50 > 25000 nM T80165 CK1I7A 71818429 IC50 = 1600 nM T80165 CH51FU 71818430 IC50 = 4000 nM T80165 CW20HQ 71818431 IC50 = 80 nM T80165 CDIR63 71818432 IC50 = 16 nM T80165 C9K3HJ 71818433 IC50 = 25 nM T80165 CFQ9C5 71818573 IC50 = 4 nM T80165 CE4K3S 71818574 IC50 = 50 nM T80165 C2L7TX 71818575 IC50 = 16 nM T80165 CPFB17 71818576 IC50 = 1600 nM T80165 CHFG76 71818577 IC50 = 63 nM T80165 CEH0X1 71818578 IC50 = 32 nM T80165 C4H6ZC 71818579 IC50 = 1260 nM T80165 CN3C5I 71818710 IC50 = 6300 nM T80165 C7TAV3 138319685 IC50 = 11 nM T80165 C81ILP 138471783 IC50 > 30000 nM T80165 CEK6B1 139300630 IC50 > 10000 nM T80165 CWJ0K6 145955642 IC50 = 280 nM T80165 CZ8W1F 145960626 IC50 = 52 nM T80165 CX3VH5 145960676 IC50 = 30 nM T80165 CJ1O5H 145961103 IC50 = 440 nM T80165 CTVR05 145961491 IC50 = 37 nM T80165 CRYN14 145961777 IC50 = 33 nM T80165 CKM9A7 145961840 IC50 = 160 nM T80165 CIM9O6 145961922 IC50 = 210 nM T80165 C0B3SG 145962010 IC50 = 500 nM T80165 CHOJ18 145962723 IC50 = 660 nM T80165 C5E3RJ 145962891 IC50 = 8 nM T80165 C6VNH3 145962956 IC50 = 22 nM T80165 C8CQX3 145963143 IC50 = 49 nM T80165 CC1T5Z 145963172 IC50 = 390 nM T80165 CWS86L 145963466 IC50 = 200 nM T80165 CF7K5G 145963483 IC50 = 3 nM T80165 CB9S3T 145963706 IC50 = 560 nM T80165 CPT8G6 155526515 IC50 = 250 nM T80165 CHNK53 155560555 IC50 = 170 nM T80165 D03LVL 53464483 IC50 > 25000 nM T19760 D03QLG 9917013 IC50 < 1 nM T19760 D06DMQ 59472121 Ki = 15 nM T19760 D0E3TC 44259 IC50 = 1.52 nM T19760 D0O6VZ 25254071 IC50 = 232 nM T19760 D03BNU 59604787 IC50 > 10000 nM T19760 D0T3ME 156422 IC50 > 30000 nM T19760 C8NW5J 3815 IC50 = 138 nM T19760 C18WEB 490561 IC50 = 22 nM T19760 CK21EQ 9796713 IC50 = 69 nM T19760 CBT0X5 9797847 IC50 = 300 nM T19760 C7JE0V 9904731 IC50 = 1415 nM T19760 CR3DA5 9939328 IC50 = 45 nM T19760 C6MO1K 10530175 IC50 = 15 nM T19760 CRJD61 10532168 IC50 = 162 nM T19760 CHB35P 10604501 IC50 = 303 nM T19760 C05KFQ 10604778 IC50 = 360 nM T19760 CJ4BN2 10626594 IC50 = 16 nM T19760 CGP93J 10745853 IC50 = 19 nM T19760 CO7Y9M 10770450 IC50 = 90 nM T19760 C7N2XF 10935867 IC50 = 308 nM T19760 CW3NL5 11012763 IC50 > 300 nM T19760 CD5I7L 11067837 IC50 = 68 nM T19760 CYXF06 11131268 IC50 = 1795 nM T19760 C85WGB 12970028 IC50 > 10000 nM T19760 CAC69O 14677298 IC50 > 10000 nM T19760 CC3J9K 15736808 IC50 = 2900 nM T19760 C20DST 16105503 IC50 = 46 nM T19760 C47EWZ 16105505 IC50 > 300 nM T19760 CSQ86L 16105506 IC50 > 300 nM T19760 C28QKT 16105508 IC50 = 482 nM T19760 CXO3N2 16105509 IC50 = 615 nM T19760 CCN62F 16105510 IC50 = 22 nM T19760 C1JXQ8 16105511 IC50 = 1106 nM T19760 C63QYN 16105513 IC50 > 300 nM T19760 CK0W9E 16105515 IC50 > 10000 nM T19760 CY8L7E 24896769 IC50 > 10000 nM T19760 C0USZ6 24971429 IC50 = 188 nM T19760 C8FK3N 24971430 IC50 = 66 nM T19760 C45WDR 24971433 IC50 = 101 nM T19760 CLPE65 24971435 IC50 = 49 nM T19760 CWP29U 25242324 IC50 = 591 nM T19760 C3E7RP 44284203 IC50 = 28 nM T19760 C8FY7N 44284204 IC50 = 43 nM T19760 CGC50I 44407533 IC50 > 1000 nM T19760 CU0H6W 44407571 IC50 > 1000 nM T19760 C3HW7L 44570553 IC50 = 5000 nM T19760 C17PVE 44570554 IC50 > 30000 nM T19760 CLOY92 44570599 IC50 = 4000 nM T19760 CK06LT 44570600 IC50 = 7000 nM T19760 CZGB46 46180666 IC50 > 1000 nM T19760 C8NA4L 53384644 IC50 > 30000 nM T19760 C8R4FE 57991377 IC50 = 370 nM T19760 C97ZGJ 58539301 IC50 = 2100 nM T19760 CT3EW2 59292007 IC50 = 51 nM T19760 CV63UL 67240318 IC50 > 10000 nM T19760 CVIA91 71553085 IC50 = 12230 nM T19760 C1TR3O 71553152 IC50 = 13430 nM T19760 CDJY72 71568837 IC50 = 370 nM T19760 CRX81Q 71575642 IC50 > 10000 nM T19760 C8CAG7 71578921 IC50 > 10000 nM T19760 CZ4BX1 72547959 IC50 = 67.8 nM T19760 CQ2OB9 90292687 IC50 = 3500 nM T19760 CHI39S 90292823 IC50 = 5920 nM T19760 CJQ5N6 91936970 IC50 > 10000 nM T19760 C5N1VZ 102581295 IC50 > 10000 nM T19760 C4X7SD 122192466 IC50 > 10000 nM T19760 CGBZ13 134843302 IC50 = 900 nM T19760 C3MK9W 136807986 IC50 > 10000 nM T19760 CXC69T 137321158 IC50 = 52 nM T19760 C6VB3O 145925651 IC50 >= 5000 nM T19760 CV9QD6 145968243 IC50 = 13 nM T19760 C2MD1Q 155513187 IC50 > 10000 nM T19760 C86HPW 155518524 IC50 = 100000 nM T19760 C68GMW 155538446 IC50 = 22000 nM T19760 CY6Q8S 155554337 IC50 = 21000 nM T19760 CO2I4P 155559898 IC50 = 600 nM T19760 D00ERW 44444843 Ki > 1667 nM T19760 D07ADX 54764565 IC50 = 19 nM T19760 D07IHM 9823787 IC50 = 33 nM T19760 D09QBA 23378546 IC50 = 103 nM T19760 D0E7VO 59627005 IC50 = 44.3 nM T19760 D0N4LR 53469448 IC50 = 1578 nM T19760 D0O6OH 71553154 IC50 = 160 nM T29728 D03LWG 53235510 IC50 > 10000 nM T29728 D0E3TC 44259 IC50 = 3370 nM T29728 C3VRO9 44557921 IC50 > 10000 nM T29728 CLS29B 46872626 IC50 > 10000 nM T29728 CV63UL 67240318 IC50 > 10000 nM T29728 C8VE2W 72695133 IC50 = 810 nM T29728 C9K7PA 72721921 IC50 = 800 nM T29728 C9HPG8 137661516 IC50 = 460 nM T29728 C2MD1Q 155513187 IC50 > 10000 nM T94201 D0U3SY 49806720 IC50 = 195 nM T94201 D0E3TC 44259 IC50 = 24.5 nM T94201 CK34LS 11632737 IC50 > 10000 nM T94201 C7YG1N 24759534 IC50 > 100000 nM T94201 CY8L7E 24896769 IC50 > 10000 nM T94201 CLS29B 46872626 IC50 > 10000 nM T94201 CXJ63M 59603829 IC50 = 28000 nM T94201 CQEU96 59603842 IC50 = 140 nM T94201 CV63UL 67240318 IC50 > 10000 nM T94201 C5DGR9 69036886 IC50 = 10000 nM T94201 C1HW4B 89735655 IC50 = 12000 nM T94201 CM1XS0 135324340 IC50 = 36 nM T94201 C2MD1Q 155513187 IC50 > 10000 nM T94201 C86HPW 155518524 IC50 = 7800 nM T94201 D00ERW 44444843 Ki = 2307 nM T94201 D0J1JB 11668217 IC50 = 40 nM T53378 D00STL 644241 Ki = 446 nM T53378 D00ZOF 23666456 Ki = 1530000 nM T53378 D01MUR 68844 IC50 = 45.3 nM T53378 D02FLB 516892 Ki = 6600000 nM T53378 D02PJA 24841 Ki = 80000 nM T53378 D02URS 4875 Ki = 80000 nM T53378 D03RTS 2662 Ki = 290 nM T53378 D03UOT 785 Ki = 10800 nM T53378 D04AIT 5280445 Ki = 293 nM T53378 D05OFX 219078 Ki = 525 nM T53378 D05UYW 5284549 Ki = 43 nM T53378 D07CWD 3657 Ki = 113000 nM T53378 D07HBX 338 Ki = 11100 nM T53378 D07INV 3295 Ki = 93 nM T53378 D07MGA 72281 Ki = 102.1 nM T53378 D07VDZ 5284627 Ki = 4900 nM T53378 D09NIA 2732 Ki = 196 nM T53378 D09VAZ 5565 Ki = 35000 nM T53378 D0AZ3C 5291 Ki = 4553 nM T53378 D0AZ8C 5213 Ki = 8960 nM T53378 D0C2II 4100 Ki = 240 nM T53378 D0C8FX 3005837 Ki = 6130 nM T53378 D0E1SW 1986 Ki = 11 nM T53378 D0E9JM 4873 Ki = 90000 nM T53378 D0H8FH 3702 Ki = 213 nM T53378 D0J4GO 3038 Ki = 95 nM T53378 D0J7RK 36811 Ki = 8980 nM T53378 D0K0OZ 5702160 Ki = 938.8 nM T53378 D0K1QD 3998 Ki = 2800 nM T53378 D0K8KX 5280343 Ki = 7890 nM T53378 D0L4JT 5333 Ki = 3000 nM T53378 D0L6DA 119607 Ki = 1340 nM T53378 D0MA7C 23668193 Ki = 30800000 nM T53378 D0OT0O 44561 Ki = 820000 nM T53378 D0PQ3G 3440 Ki = 564 nM T53378 D0SH3I 387447 Ki = 6510 nM T53378 D0U5QK 1983 Ki = 11400 nM T53378 D0Y2IZ 5560 Ki = 449 nM T53378 D0Z3EI 6038 Ki = 360 nM T53378 D0Z4UY 517045 Ki = 550000 nM T53378 D02ECG 23662274 Ki = 14500 nM T53378 D04PBH 5280804 Ki = 75.7 nM T53378 D05NJI 5287541 Ki = 24 nM T53378 D08BXT 1102 Ki = 112 nM T53378 D0I7MT 5281807 Ki > 10000 nM T53378 D0L6HN 996 Ki = 9500 nM T53378 D0SC6I 517055 Ki = 74700 nM T53378 D0U3EP 445154 Ki = 4470 nM T53378 D0V0UK 82267 Ki = 880 nM T53378 D03SLR 445858 Ki = 10800 nM T53378 D0NH9P 135 Ki = 7780 nM T53378 D0X2AU 23427 Ki > 100000 nM T53378 D0LD9S 1103 Ki = 10 nM T53378 CI0WH9 72 Ki = 2450 nM T53378 CUT2V4 260 Ki = 90000 nM T53378 COV5W3 402 Ki = 3900000 nM T53378 CSZ43B 540 Ki = 610000 nM T53378 C97QXH 767 Ki = 5700000 nM T53378 C39CTO 768 Ki = 770000 nM T53378 C1QDT0 781 Ki = 39000000 nM T53378 CAD4R0 798 Ki = 2330 nM T53378 CW0R2L 944 Ki = 58700000 nM T53378 C2LNM9 1016 Ki = 3180000 nM T53378 CQV86E 1100 Ki = 13200000 nM T53378 C8W7BZ 1118 Ki = 9000000 nM T53378 CU12QE 1203 Ki = 4900 nM T53378 C5L7VX 2871 Ki = 5480 nM T53378 CZP5J2 3415 Ki = 820000 nM T53378 CJ2F6P 5056 Ki = 4010 nM T53378 CDJ4K6 5987 Ki = 930 nM T53378 CU9EM3 6125 Ki = 99 nM T53378 CUP2F4 7043 Ki = 14320 nM T53378 C1CVT7 7121 Ki = 6480 nM T53378 C6NC4O 7414 Ki = 8100 nM T53378 CIU0C8 7519 Ki = 14320 nM T53378 CXF7C6 8736 Ki = 53700 nM T53378 CR3IF4 8865 Ki = 2800 nM T53378 COU60V 10340 Ki = 5700000 nM T53378 CUG8B9 11418 Ki = 8430 nM T53378 CCPT31 11419 Ki = 8930 nM T53378 C57OTC 13818 Ki = 310000 nM T53378 CKA21F 14768 Ki = 2150000 nM T53378 CUA0L6 14917 Ki = 70000 nM T53378 CS8X0P 16124 Ki = 5340000 nM T53378 CS39YR 19654 Ki = 64900000 nM T53378 CF14KR 24247 Ki = 767000000 nM T53378 C4IZB8 24345 Ki = 108700000 nM T53378 C9M8EJ 24434 Ki = 58700000 nM T53378 CAN29U 24436 Ki = 9000000 nM T53378 C8S9AF 24445 Ki = 128000000 nM T53378 C3NG2U 24529 Ki = 30800000 nM T53378 CFM9L6 24530 Ki = 65100000 nM T53378 C3F1OY 25502 Ki = 640000 nM T53378 C7YZM4 33557 Ki = 65100000 nM T53378 C4OU6D 35703 Ki = 35700 nM T53378 C89DPG 39981 Ki = 79 nM T53378 CY2GU3 60582 Ki = 486 nM T53378 C1N6SE 61127 Ki = 17480 nM T53378 CF26VS 61441 Ki = 27500000 nM T53378 CLMR98 61857 Ki = 17400000 nM T53378 C6DG9Q 65185 Ki = 226000000 nM T53378 CE5RZ1 76509 Ki = 53 nM T53378 CX79KD 78297 Ki = 885.3 nM T53378 CX47BZ 78479 Ki = 44000 nM T53378 CJ01AO 94706 Ki = 15 nM T53378 C1GQE3 97576 Ki = 4450 nM T53378 CEC01M 97598 Ki = 4736 nM T53378 C6K3MG 101424 Ki > 100000 nM T53378 CDP5M6 125623 Ki = 234 nM T53378 CN19UT 129695 Ki = 18 nM T53378 CUX39B 132037 Ki = 1840 nM T53378 CCK5Y6 133125 Ki = 6.7 nM T53378 CD2HC7 138614 Ki = 8670 nM T53378 C2P0RH 139584 Ki = 920000 nM T53378 C6M0TK 167985 Ki = 97000000 nM T53378 C7DS2I 228958 Ki = 83 nM T53378 C0B3OQ 253877 Ki = 90000 nM T53378 C1QOB5 284045 Ki = 145120 nM T53378 C96DKW 310360 Ki = 286 nM T53378 CT3ZU4 388776 Ki = 116 nM T53378 CH21KA 389641 Ki = 104000 nM T53378 C6CQO3 389642 Ki = 103000 nM T53378 CNPZ40 394897 Ki = 349 nM T53378 C7HME8 439246 Ki = 79.5 nM T53378 C5HM8E 474578 Ki = 675.3 nM T53378 COGF52 516871 Ki = 39000000 nM T53378 C5OA7L 522689 Ki = 70000 nM T53378 CJ7FR6 533728 Ki = 6500 nM T53378 C8J7CO 730546 Ki = 4797 nM T53378 C6T0NU 1230924 Ki = 280.5 nM T53378 C40CKN 1316238 Ki = 7109 nM T53378 C6FN0O 2316976 Ki = 9578 nM T53378 C4TD8M 2388085 Ki = 449.4 nM T53378 CKH53Q 2723810 Ki = 1250000 nM T53378 C8QGL9 2760606 Ki > 10000 nM T53378 CNGK51 2781602 Ki = 175 nM T53378 C21FUI 2801263 Ki = 1430 nM T53378 CE2GR3 2900806 Ki = 12300 nM T53378 CJ9LZ7 3051101 Ki = 76.4 nM T53378 C6V3ES 3365615 Ki = 28 nM T53378 C86GSL 3542746 Ki = 37 nM T53378 CD0FL4 3627258 Ki = 52 nM T53378 CV0KG3 3950536 Ki > 10000 nM T53378 C37ZWJ 4369171 IC50 = 7.41 nM T53378 C0PX7R 4369172 IC50 = 4.25 nM T53378 CDK4L0 4608376 Ki = 290000 nM T53378 C07MRI 4712722 Ki = 500000 nM T53378 CUA65R 4857564 Ki = 8365 nM T53378 CN31CX 5071527 Ki = 156 nM T53378 C7GXU1 5147921 Ki = 19100000 nM T53378 C4HB1G 5172319 Ki = 7 nM T53378 CI8JY0 5172475 Ki = 355 nM T53378 CEN0L7 5227639 Ki = 41 nM T53378 CEBD92 5272990 Ki = 6200 nM T53378 CP09FG 5272997 Ki = 26600 nM T53378 CN10FM 5281793 Ki = 66.6 nM T53378 CH5OM1 5463917 Ki = 44800000 nM T53378 C9L8AX 6537802 Ki = 750 nM T53378 C65FRB 6852128 Ki = 146 nM T53378 CKCM96 7463376 Ki = 3910 nM T53378 CDCP43 7766335 Ki = 39500 nM T53378 CNKD31 10016330 Ki = 853.6 nM T53378 CGU6P4 10021113 IC50 = 128 nM T53378 C5X7GY 10059582 Ki = 1427 nM T53378 CWM01R 10059806 Ki = 7640 nM T53378 C0P5XV 10081897 Ki = 896.6 nM T53378 CD58EL 10083644 Ki = 18700 nM T53378 C7WU0A 10107532 Ki = 1557 nM T53378 CXD91O 10136406 Ki = 6028 nM T53378 CJV68L 10220266 Ki = 1031 nM T53378 CM4E8G 10243877 Ki = 125 nM T53378 CQ8A0I 10328097 Ki = 62.2 nM T53378 CN40WD 10331524 Ki = 1748 nM T53378 C58IYR 10366827 Ki = 1080 nM T53378 C3HBY6 10375558 Ki = 450 nM T53378 CVIN94 10439991 Ki = 344.2 nM T53378 CD41CA 10512636 Ki > 10000 nM T53378 CWQY26 10535227 Ki > 10000 nM T53378 C73KXU 10586607 Ki = 9100 nM T53378 C9TSQ6 10632698 Ki = 31300 nM T53378 C6D2TJ 10712038 Ki = 941 nM T53378 CPN13K 10864662 Ki = 265 nM T53378 C8OKX5 10865717 Ki = 6 nM T53378 C1LX6K 10887220 Ki = 27 nM T53378 CKL08U 10897133 Ki = 190 nM T53378 CWGB92 10907843 Ki = 40 nM T53378 C6EPH9 10919571 Ki = 425 nM T53378 CTDR05 10920174 Ki = 25 nM T53378 CVR31W 10930187 Ki = 27 nM T53378 C5ZPE9 10963315 Ki = 5 nM T53378 C3IDH7 10974944 Ki = 21 nM T53378 C8JAX5 10996222 Ki = 430 nM T53378 C60TSD 10996432 Ki = 5 nM T53378 CNCX57 11017060 Ki = 500 nM T53378 C4WU6R 11017835 Ki = 29 nM T53378 C5CJU7 11028005 Ki = 550 nM T53378 CLM10Q 11028999 Ki = 18 nM T53378 C36BAC 11034581 Ki > 100000 nM T53378 COA8S5 11039158 Ki = 32 nM T53378 CL46GE 11039314 Ki = 6 nM T53378 CT2D9I 11060771 Ki = 630 nM T53378 C6FA8Y 11060833 Ki = 19 nM T53378 C5X4DW 11060882 Ki = 36 nM T53378 C8C6ER 11069133 Ki = 15 nM T53378 CIAW06 11082579 Ki = 9 nM T53378 C3O5JB 11083515 Ki = 4 nM T53378 CYST27 11093710 Ki = 36 nM T53378 CMK4Y0 11096006 Ki = 708.6 nM T53378 CYQ01S 11115351 Ki = 25 nM T53378 C25CRH 11146161 Ki = 29 nM T53378 CO6X8J 11147037 Ki = 9 nM T53378 CIL4M9 11183499 Ki > 100000 nM T53378 C39IDU 11183936 Ki = 4627 nM T53378 CHC42Y 11245700 Ki = 842 nM T53378 CF15AS 11287957 Ki = 76.1 nM T53378 CA6T0Z 11322287 Ki = 4442 nM T53378 CXB86F 11579563 Ki = 4215 nM T53378 C9QL2F 11615432 Ki = 3459 nM T53378 CDU79V 11637531 Ki = 5726 nM T53378 CX4W3J 11701693 Ki = 4082 nM T53378 CEGC64 11735346 Ki = 115 nM T53378 CX5LA8 11763331 Ki = 180 nM T53378 CV7HN1 11795548 Ki = 60 nM T53378 C18JIA 11828627 Ki = 330 nM T53378 CE71FU 11828964 Ki = 8 nM T53378 CJRD82 11966600 Ki = 16 nM T53378 CXSE37 11967046 Ki = 170 nM T53378 C9VM6I 11967472 Ki = 24 nM T53378 CQXG94 11970596 Ki = 9900 nM T53378 C4ZYQ1 12049713 Ki = 1690000 nM T53378 CMPA32 12066940 Ki > 500000 nM T53378 CB15KR 12066941 Ki = 309000 nM T53378 CREV05 12140130 Ki = 4573 nM T53378 C5RS4H 12528487 Ki = 1228 nM T53378 CM8TP6 12528490 Ki = 1945 nM T53378 CC25BI 13927398 Ki = 850000 nM T53378 C7K4JV 14024589 Ki = 3894 nM T53378 CNZ6H2 14205726 Ki = 5500000 nM T53378 C92OEB 14498136 Ki = 218.1 nM T53378 CHOG93 14611919 Ki = 9000 nM T53378 CK8GE9 15230629 Ki = 2692 nM T53378 CLT47Z 15783680 Ki = 69.2 nM T53378 C8PER5 15938557 Ki > 500000 nM T53378 C3W2MB 15939939 Ki = 67.3 nM T53378 CC0Z4V 16119626 Ki = 9670 nM T53378 CG7OL3 16693908 Ki = 124000000 nM T53378 CK7D2I 17748220 Ki = 43700 nM T53378 C3AX8E 17774014 Ki = 5461 nM T53378 C6SFI8 18268734 Ki = 9657 nM T53378 C61KUX 21726402 Ki = 75.3 nM T53378 C54IUM 21778115 Ki = 28040 nM T53378 C27BJH 21778117 Ki = 27480 nM T53378 C9U4TE 22313850 Ki = 9540 nM T53378 CICR37 23426698 Ki = 45740 nM T53378 C1Y2JB 24286289 Ki = 179.3 nM T53378 C8BL9O 24762836 Ki = 9610 nM T53378 CQG9O0 24816432 Ki = 47 nM T53378 COI25U 25131351 Ki = 44 nM T53378 CNMY17 25131685 Ki = 345 nM T53378 CG0S7T 25154732 Ki = 8760 nM T53378 CYG1H9 25154741 Ki = 10050 nM T53378 CPN2T5 25392418 Ki = 8012 nM T53378 CLNR46 26598995 Ki = 5885 nM T53378 CBPO08 34751720 Ki = 2940.3 nM T53378 C82MRL 44144383 Ki = 48.9 nM T53378 CMR52W 44201382 IC50 = 64 nM T53378 CIG89O 44201383 IC50 = 246 nM T53378 CI3O9B 44395149 Ki = 704 nM T53378 CZ4DF9 44399462 Ki = 97 nM T53378 CD5MJ6 44399571 Ki = 89 nM T53378 C2T7MB 44399654 Ki = 8620 nM T53378 CM3J0U 44430517 Ki = 850 nM T53378 C9LT7Y 44430518 Ki = 10 nM T53378 C1VTB6 44430520 Ki = 30700 nM T53378 C2L5MB 44430521 Ki = 1040 nM T53378 CVEO17 44430523 Ki = 670 nM T53378 C8MFL1 44430524 Ki = 89300 nM T53378 C8E0MV 44552472 Ki = 1032 nM T53378 CKG53H 44552473 Ki = 543 nM T53378 C17XAJ 44552559 Ki = 435 nM T53378 CJ05ZA 44571847 Ki = 4320 nM T53378 C52WIF 44571892 Ki = 6100 nM T53378 COE8U0 45267045 Ki = 65.6 nM T53378 C23MVW 45269009 IC50 = 380 nM T53378 C0RG8K 45269749 Ki = 7100 nM T53378 CJX37G 45375967 Ki = 4360 nM T53378 CJ68EO 45375968 Ki = 181 nM T53378 CSE48D 45375973 Ki = 3905 nM T53378 CV5RQ3 45484187 Ki = 3800 nM T53378 CTG20B 45485271 Ki = 11800 nM T53378 CK4U0V 45485283 Ki > 500000 nM T53378 CW7FR9 45486144 Ki = 46 nM T53378 C8T4WM 45486167 Ki = 339 nM T53378 CHE08Y 46225608 Ki = 4852 nM T53378 CIE2H3 46225609 Ki = 5341 nM T53378 CF42NR 46225631 Ki = 617 nM T53378 C0ZG3L 46225639 Ki = 778 nM T53378 CGW1I5 46225644 Ki = 532 nM T53378 CEOQ06 46225645 Ki = 875 nM T53378 CR0WO3 46225646 Ki = 912 nM T53378 CC2BL5 46225656 Ki = 943 nM T53378 CW52PZ 46225672 Ki = 842 nM T53378 CXJ1C9 46225673 Ki = 765 nM T53378 CQN8K4 46635132 Ki = 1780 nM T53378 C2RA7G 46861342 Ki = 1495 nM T53378 CCW34G 46861804 IC50 = 33.1 nM T53378 CRZ29M 46861805 IC50 = 1890 nM T53378 CI21XG 46861806 IC50 = 188 nM T53378 CT65RE 46868356 Ki = 494.4 nM T53378 CT9OQ6 46887904 IC50 = 241 nM T53378 CVX05D 46887935 IC50 = 575 nM T53378 CZ23PM 46887936 IC50 = 2040 nM T53378 C6QT5B 46887937 IC50 = 1480 nM T53378 CTL5J9 46887938 IC50 = 952 nM T53378 CNT04P 46887939 IC50 > 5000 nM T53378 C6EZM9 46887969 IC50 = 783 nM T53378 CTM4O2 46887970 IC50 = 1910 nM T53378 CCGD62 46887971 IC50 > 5000 nM T53378 CBMK80 46887972 IC50 > 5000 nM T53378 C2Z0FD 46887973 IC50 = 1450 nM T53378 C1BW9J 46887974 IC50 = 283 nM T53378 C9KMN4 46888010 IC50 > 5000 nM T53378 C52NDI 46888011 IC50 = 361 nM T53378 C5H0YK 46888012 IC50 = 229 nM T53378 CP0O7K 46888057 IC50 = 23 nM T53378 C6TXO0 46888058 IC50 = 126 nM T53378 CVU6W4 46888059 IC50 = 46.8 nM T53378 C53URE 46888060 IC50 = 118 nM T53378 CIC14R 46888061 IC50 = 23 nM T53378 CS0J9F 46888093 IC50 = 139 nM T53378 C51JUC 46888094 IC50 = 20.9 nM T53378 C7W2QG 46888095 IC50 = 23 nM T53378 CV49AY 46888096 IC50 = 1230 nM T53378 CEAQ12 46888136 IC50 = 402 nM T53378 CLT61J 46888137 IC50 = 2660 nM T53378 CFLG09 46888138 IC50 = 2190 nM T53378 C5I0CN 46888139 IC50 = 1250 nM T53378 C93AIR 46899573 Ki = 108000 nM T53378 CJ0R2O 46911381 Ki = 413 nM T53378 CPGW70 53245686 Ki = 154 nM T53378 CF89ML 53307609 Ki = 32720 nM T53378 C0NUM6 53386724 Ki = 7200 nM T53378 C54FGU 53386866 Ki = 6740 nM T53378 CRI54V 53386867 Ki = 7450 nM T53378 CUX7S4 53386868 Ki = 7500 nM T53378 CHCT45 54580732 Ki = 76 nM T53378 CYB47X 54581736 Ki = 38 nM T53378 CW2KI4 54582723 Ki = 46 nM T53378 CWK6B0 54582724 Ki = 89 nM T53378 CBS8R1 54584666 Ki = 225 nM T53378 CJ3UE2 54584667 Ki = 139 nM T53378 CO0BD9 54585508 Ki = 148 nM T53378 C0A5OZ 54612935 Ki = 653.2 nM T53378 C3RQX8 54940826 Ki = 4849 nM T53378 C2UE8F 56682961 Ki = 16 nM T53378 CIJ9V0 56684131 Ki = 7500 nM T53378 CH52DA 56921864 Ki = 3600 nM T53378 CUR32K 57334711 Ki = 850 nM T53378 C2CD1R 57334712 Ki = 870 nM T53378 C1K0DM 57334713 Ki = 880 nM T53378 CP7YR5 57345662 Ki = 260 nM T53378 C87ASQ 57387395 Ki = 47.2 nM T53378 C13FJU 57392368 Ki = 930 nM T53378 CY5G4Z 57395885 Ki = 1120 nM T53378 C5RX6H 57396029 Ki = 7420 nM T53378 CP75OF 57397664 Ki = 46350 nM T53378 CUAG84 57397836 Ki = 102400 nM T53378 CW43HV 57397837 Ki = 7680 nM T53378 C1MCW8 57399336 Ki = 48730 nM T53378 C2CAM1 57399491 Ki = 7030 nM T53378 CG3W0D 58404071 Ki = 1420 nM T53378 C2J7GW 66572313 Ki = 42260 nM T53378 C7J5RN 66573254 Ki = 57610 nM T53378 CRHL03 70689373 Ki = 5 nM T53378 CQR91N 70692438 Ki = 30780 nM T53378 CWJ0Q8 70696540 Ki = 13120 nM T53378 C8NYL3 71449075 Ki = 21 nM T53378 CXJ16H 71450117 Ki = 328 nM T53378 CK04AG 71450862 Ki = 4 nM T53378 CB8JA3 71455488 Ki = 7140 nM T53378 C02UHX 71455489 Ki = 8850 nM T53378 CICJ97 71457274 Ki = 7200 nM T53378 CX9KJ3 71459903 Ki = 100 nM T53378 CMHG14 71521493 Ki = 4900 nM T53378 CHN53G 71521494 Ki = 7800 nM T53378 CZJ5M6 71521495 Ki = 6700 nM T53378 CFBE53 71521496 Ki = 8300 nM T53378 CME27W 71521497 Ki = 9200 nM T53378 C24XWU 71521575 Ki = 5600 nM T53378 CJF68W 71521576 Ki = 8400 nM T53378 C7NMJ2 71714066 Ki = 4120 nM T53378 C5DEF6 71714067 Ki = 13700 nM T53378 C50LSJ 71714068 Ki = 5360 nM T53378 C0ROQ1 71770179 Ki = 9232 nM T53378 C63MIX 72163344 Ki = 8839 nM T53378 C3UJ8A 72695827 Ki = 717.7 nM T53378 CX82JD 72696463 Ki = 717 nM T53378 COCV73 72696591 Ki = 1360 nM T53378 C5KHD7 72696592 Ki = 2552 nM T53378 C4FBA6 72696593 Ki = 603 nM T53378 CO1JM5 72696594 Ki = 2744 nM T53378 CUF61Q 72696595 Ki = 3660 nM T53378 CO1JT3 73054728 Ki = 627 nM T53378 CZ5X4W 76328576 Ki = 8175 nM T53378 CU9I6V 82078731 Ki = 461 nM T53378 C5TB6O 82080973 Ki = 1637 nM T53378 C6UZR9 82911195 Ki = 1734.8 nM T53378 C6HC8V 86692720 Ki = 370.8 nM T53378 C0CR6D 90681501 Ki = 4790 nM T53378 C3AYZ5 91811067 Ki = 379.8 nM T53378 C28QRZ 101564149 Ki > 100000 nM T53378 CDGZ03 101879106 Ki = 438.95 nM T53378 CY6ER7 101879108 Ki = 737.69 nM T53378 CB1PK8 102151146 Ki = 23500 nM T53378 C0A6FY 102151151 Ki > 100000 nM T53378 C1XV9H 102311866 Ki > 100000 nM T53378 C0CVO4 102480165 Ki > 100000 nM T53378 CKV43U 118710106 Ki = 9726 nM T53378 CBAQ59 118710108 Ki = 8142 nM T53378 C0D1SQ 118724328 Ki = 233.19 nM T53378 C89YTC 118724329 Ki = 879.8 nM T53378 CBT87C 118724330 Ki = 779.7 nM T53378 C49AWZ 118724331 Ki = 397.89 nM T53378 CE3IV5 118729477 Ki = 1621.7 nM T53378 CUQ7H9 119082247 Ki = 298.4 nM T53378 CH1N0C 122193189 Ki = 24100 nM T53378 C19HVL 122193190 Ki = 33200 nM T53378 C5TQJ1 122193251 Ki = 40500 nM T53378 C8XCL0 122193252 Ki = 12500 nM T53378 CC1UO6 122226187 Ki = 52400 nM T53378 C7T0FH 122226188 Ki = 9100 nM T53378 C3EG2B 122226189 Ki = 56800 nM T53378 C26IUP 122386532 Ki > 100000 nM T53378 CY1JU3 127037755 Ki > 10000 nM T53378 C0UQ7W 127037756 Ki > 10000 nM T53378 CQUE67 127037757 Ki = 526.7 nM T53378 CG8B3V 127039153 Ki = 184.4 nM T53378 CIO74C 127039154 Ki = 72.7 nM T53378 C0L8NH 127039155 Ki = 495.6 nM T53378 CS96GU 127039479 Ki = 366.4 nM T53378 C3J8ET 127040041 Ki > 10000 nM T53378 CQC6A4 127042329 Ki = 891.9 nM T53378 C5EX6R 127048632 Ki = 400.4 nM T53378 CK1X5H 127048994 Ki = 29.7 nM T53378 C2XK0I 127048995 Ki = 29.8 nM T53378 CY4P2X 127048996 Ki = 60.6 nM T53378 C6JB5S 127048997 Ki = 708 nM T53378 CP40EB 127049242 Ki = 4.4 nM T53378 CLFB54 127049248 Ki = 5.8 nM T53378 C1T3WG 127049310 Ki = 361 nM T53378 CKO03S 127049970 Ki = 358.5 nM T53378 CP8KG9 127049971 Ki = 73.8 nM T53378 C9EJ6L 127050230 Ki = 248.3 nM T53378 C7MI5Q 127050568 Ki = 403.8 nM T53378 C1RGQ6 127050569 Ki = 138.6 nM T53378 CB5W0L 127050570 Ki = 131.6 nM T53378 CUG58A 127050571 Ki = 425.6 nM T53378 CG17IO 127050812 Ki = 9.5 nM T53378 C8X6CY 127050822 Ki = 5.5 nM T53378 C9FZ4E 127050900 Ki = 96.1 nM T53378 C4IA5N 127051119 Ki = 7.8 nM T53378 CRDQ30 127051120 Ki = 5 nM T53378 CUWE95 127051804 Ki = 378.2 nM T53378 COBU26 127051805 Ki = 519.9 nM T53378 C7SIY6 127051806 Ki = 425.4 nM T53378 C5Y4DI 127051953 Ki = 6.4 nM T53378 CJ7WT3 127052106 Ki = 466.7 nM T53378 C26TUM 127052712 Ki = 62.7 nM T53378 C7PS8D 127052713 Ki = 340.2 nM T53378 C32ART 127052714 Ki = 436 nM T53378 C9D6CB 127053004 Ki = 283.1 nM T53378 CJC35Q 129856021 Ki = 48.3 nM T53378 CCF61S 129883275 Ki = 4375 nM T53378 CNB2M7 131839635 Ki = 1782 nM T53378 CXN16P 132495328 Ki = 44.1 nM T53378 C5O1JE 132547793 Ki > 100000 nM T53378 CKYC42 132547798 Ki > 100000 nM T53378 C7MZ8T 132569639 Ki = 3000 nM T53378 C4K1YW 132961363 Ki = 94.1 nM T53378 CQ64ZM 132961364 Ki = 8.9 nM T53378 C5LGV6 132961365 Ki = 207.2 nM T53378 CD9ET2 132961426 Ki = 973 nM T53378 CR80OW 132961427 Ki = 8517 nM T53378 C2AIR8 134129901 Ki = 34.7 nM T53378 C1Y9AL 134130029 Ki = 7.4 nM T53378 CU10DE 134130177 Ki = 1.8 nM T53378 CP8XK0 134130364 Ki = 0.65 nM T53378 C83LZE 134130471 Ki = 0.64 nM T53378 C5N8AO 134130483 Ki = 47 nM T53378 C9V3LX 134130512 Ki = 51 nM T53378 CO7G6J 134130566 Ki = 43.1 nM T53378 C69IZA 134130639 Ki > 10000 nM T53378 C8MGN3 134130817 Ki = 372.3 nM T53378 C52IRH 134131086 Ki = 0.95 nM T53378 C9HVL2 134131189 Ki = 0.53 nM T53378 C7GBW5 134131361 Ki = 35.5 nM T53378 C3WJR8 134131535 Ki = 5 nM T53378 CQ0K5P 134131567 Ki = 34.7 nM T53378 C8Q5JZ 134131574 Ki = 3.7 nM T53378 CZQ3T2 134132041 Ki > 10000 nM T53378 C89TVU 134132755 Ki = 311.8 nM T53378 CFQG76 134133776 Ki = 407 nM T53378 CT8Z2Q 134133785 Ki = 286.2 nM T53378 CHR23F 134137004 Ki > 10000 nM T53378 C2X1UG 134137145 Ki = 145.5 nM T53378 CHM19B 134139215 Ki = 108 nM T53378 CRNF42 134140829 Ki = 197.6 nM T53378 C1T9JU 134140936 Ki = 7345 nM T53378 CG4NU1 134141378 Ki = 266 nM T53378 CIK25S 134142323 Ki = 71.3 nM T53378 CIRG86 134142877 Ki = 47.2 nM T53378 CWT6O9 134142989 Ki = 113.4 nM T53378 C5BD1C 134143174 Ki > 10000 nM T53378 CWQ62J 134144541 Ki = 4429.4 nM T53378 CG7X9K 134144756 Ki = 6056 nM T53378 CJ5QD3 134144926 Ki = 428.4 nM T53378 CR5F8T 134145685 Ki = 410.4 nM T53378 C8FV5Y 134147016 Ki > 10000 nM T53378 C0TV9S 134147261 Ki = 8489 nM T53378 C85ABV 134147911 Ki = 79.6 nM T53378 CGBZ05 134148709 Ki = 2791 nM T53378 CS7K8C 134149271 Ki = 443.8 nM T53378 CD5TI1 134149815 Ki = 2396.8 nM T53378 CZ2C3J 134149835 Ki = 2485 nM T53378 CIL4H9 134151823 Ki > 10000 nM T53378 C9GF7L 134152087 Ki = 451.3 nM T53378 CZ4WI8 134152920 Ki = 288.1 nM T53378 CD4EN0 134153199 Ki = 7301 nM T53378 CH6OT4 134153506 Ki = 442.3 nM T53378 CZ9T6I 134153525 Ki > 10000 nM T53378 CWSI54 134154346 Ki = 292.9 nM T53378 CQZU97 134154945 Ki > 10000 nM T53378 C52UTP 134156470 Ki = 246.2 nM T53378 C7OV6T 134156655 Ki = 304.5 nM T53378 CZ9L5F 134158397 Ki = 66.8 nM T53378 C8C0TO 134812637 Ki = 2246.9 nM T53378 CV9X5Y 134817795 Ki = 4.6 nM T53378 CW9B7C 135422576 Ki = 348.3 nM T53378 CPW4T3 135530880 Ki = 36.6 nM T53378 CYKW91 136728963 Ki = 272.3 nM T53378 CZ5GQ4 137631746 Ki = 9.8 nM T53378 C83VZC 137632115 Ki = 200 nM T53378 CBJ75C 137632178 Ki = 2069.5 nM T53378 CL5K3D 137632743 Ki = 5.6 nM T53378 C5J3AX 137633409 Ki = 4 nM T53378 C5NLG4 137634142 Ki = 2980 nM T53378 C7N0ER 137634525 Ki > 100000 nM T53378 C29PFJ 137634549 Ki = 3960 nM T53378 CP0EC3 137635051 Ki = 6148 nM T53378 C08ANJ 137635055 Ki = 2920 nM T53378 C3NQ9Y 137635300 Ki = 9391 nM T53378 CZ1O5K 137635430 Ki = 4620 nM T53378 CV12YX 137636350 Ki = 0.79 nM T53378 CLR6U5 137636505 Ki = 9358 nM T53378 C5D3BS 137636775 Ki = 3560 nM T53378 C0H2CK 137637173 Ki = 184.5 nM T53378 CWO5Z6 137637365 Ki = 8.8 nM T53378 C80KCO 137637736 Ki = 40.7 nM T53378 CHQ3P9 137638456 Ki = 16.3 nM T53378 COE61G 137639833 Ki = 78900 nM T53378 CZGW35 137640627 Ki = 4700 nM T53378 C53ZAF 137641717 Ki > 10000 nM T53378 CR5JZ8 137642047 Ki > 10000 nM T53378 CCSN50 137642054 Ki = 8.3 nM T53378 C6YV7B 137642310 Ki = 4250 nM T53378 C61TSP 137642864 Ki > 100000 nM T53378 C1BW5I 137643671 Ki > 100000 nM T53378 CN2M3C 137643724 Ki = 2520 nM T53378 C0B8QA 137643949 Ki = 0.73 nM T53378 CF31BQ 137644307 Ki = 79.4 nM T53378 CI4A9L 137644641 Ki = 4900 nM T53378 CFA3R0 137644914 Ki = 44.7 nM T53378 CHG72J 137644957 Ki = 2925 nM T53378 CDZ6T8 137645734 Ki = 329.3 nM T53378 C4WOE0 137646284 Ki = 9380 nM T53378 C0YFX2 137646956 Ki > 10000 nM T53378 CRP78K 137647221 Ki = 4.4 nM T53378 C49PLO 137648279 Ki = 1433.5 nM T53378 C21TVD 137648644 Ki > 10000 nM T53378 C6RIM2 137648717 Ki = 36.3 nM T53378 CEZT03 137649001 Ki = 530.5 nM T53378 CI9LS2 137649321 Ki = 46.1 nM T53378 CY94BR 137649373 Ki = 2230 nM T53378 CD7S5L 137650698 Ki > 100000 nM T53378 CJV8Q6 137650823 Ki = 912 nM T53378 CV89IF 137651491 Ki = 26.6 nM T53378 C01BXO 137651769 Ki = 2.6 nM T53378 CY0C6Z 137652226 Ki = 9.5 nM T53378 C6GWB1 137652305 Ki = 9 nM T53378 CN3RQ8 137652373 Ki > 10000 nM T53378 CP4GY0 137652940 Ki = 4330 nM T53378 C03TAW 137653117 Ki = 3580 nM T53378 CTP0U2 137654343 Ki = 31.2 nM T53378 CS3LD8 137654917 Ki = 2450 nM T53378 CXC7I2 137655261 Ki = 42.8 nM T53378 C3DT7S 137655450 Ki = 9.4 nM T53378 CASB61 137655528 Ki = 0.81 nM T53378 CC0OY9 137655984 Ki = 33.1 nM T53378 C8TJN9 137656061 Ki = 1752 nM T53378 COEY05 137656447 Ki = 36.7 nM T53378 C0CK7G 137656796 Ki = 1799.5 nM T53378 C8RNZ6 137657759 Ki = 9.1 nM T53378 CT5PO9 137658239 Ki = 3560 nM T53378 C3W4BA 137658271 Ki = 6764 nM T53378 C41MLN 137658275 Ki > 10000 nM T53378 CL2H0T 137658375 Ki = 9.1 nM T53378 CT98MV 137658877 Ki = 0.44 nM T53378 CXO9Y7 137659205 Ki = 7.5 nM T53378 CO1RD4 137659342 Ki = 3010 nM T53378 C5AM2K 137659383 Ki > 10000 nM T53378 C60DEN 137660288 Ki = 9.3 nM T53378 C0TZD5 137661006 Ki > 100000 nM T53378 C0PIE6 137661027 Ki = 533.4 nM T53378 CQ56MJ 137661167 Ki = 270.2 nM T53378 CMP8S7 137662201 Ki = 7.5 nM T53378 CFR73V 137662256 Ki > 10000 nM T53378 CIX41M 138393379 Ki = 627 nM T53378 C7V9ZF 138455154 Ki = 326.2 nM T53378 CBOM51 138753317 Ki = 96.6 nM T53378 CQC2D5 145949182 Ki = 29.3 nM T53378 C0Z2WP 145949184 Ki = 2.6 nM T53378 CK65AC 145949290 Ki = 1164.6 nM T53378 C8BZI0 145949366 Ki = 1826.6 nM T53378 CHVR98 145949393 Ki = 8133 nM T53378 C3LZH7 145949437 Ki = 469.6 nM T53378 C09ZGW 145949615 Ki = 3347 nM T53378 CA01QK 145949650 Ki = 3.6 nM T53378 C7I3GC 145949670 Ki = 2255.5 nM T53378 CIU2Y1 145949743 Ki = 341.1 nM T53378 CA05JL 145949806 Ki = 87.7 nM T53378 CHI5L3 145949836 Ki = 5.4 nM T53378 C3U1AB 145949909 Ki = 294.7 nM T53378 C20RXT 145949974 Ki = 377.7 nM T53378 CJ8R3M 145950033 Ki = 66.9 nM T53378 CISR74 145950124 Ki = 7.8 nM T53378 CO9UN4 145950340 Ki = 618.1 nM T53378 CW56LV 145950373 Ki = 73 nM T53378 C0C9FT 145950755 Ki = 2009.2 nM T53378 CRD27H 145950965 Ki = 2 nM T53378 C9QUL0 145951028 Ki = 2321 nM T53378 C7W5PI 145951214 Ki = 79.4 nM T53378 C7LMU1 145951380 Ki = 68 nM T53378 C86DBE 145951463 Ki = 3912.1 nM T53378 CB8V7M 145951488 Ki = 772.5 nM T53378 C38QHU 145951654 Ki = 961.2 nM T53378 CIM8X0 145951670 Ki = 319.3 nM T53378 CH9J8K 145951685 Ki = 73.3 nM T53378 C74RDJ 145951698 Ki = 555.7 nM T53378 CJ2W6V 145951720 Ki = 33.4 nM T53378 CZ23SB 145951758 Ki = 4166.8 nM T53378 CC0P1U 145951787 Ki = 311.1 nM T53378 CF20QP 145951819 Ki = 8.7 nM T53378 C98SYV 145951855 Ki = 299.5 nM T53378 CF7U3J 145951902 Ki = 709.5 nM T53378 C4N3QL 145952239 Ki = 458.2 nM T53378 CP92AH 145952604 Ki = 912 nM T53378 C81UYG 145952794 Ki = 5.6 nM T53378 C6PZ3H 145952834 Ki = 914.4 nM T53378 CK4Q0X 145952846 Ki = 213.7 nM T53378 C56QVF 145952880 Ki = 429.2 nM T53378 CAS8M7 145952940 Ki = 2296 nM T53378 C5C9RI 145953173 Ki = 2646.9 nM T53378 CQM0J4 145953285 Ki = 5.1 nM T53378 C5DJY9 145953324 Ki = 2825 nM T53378 CZO1Y8 145953466 Ki = 84.9 nM T53378 CFW94A 145953493 Ki = 78 nM T53378 C80OQZ 145953572 Ki = 95.8 nM T53378 C36ENH 145953837 Ki = 7.1 nM T53378 CH9N6D 145954010 Ki = 277.4 nM T53378 CD52IH 145954185 Ki = 608.2 nM T53378 C7LZ1G 145954524 Ki = 3122.9 nM T53378 CZG7I4 145954697 Ki = 79.7 nM T53378 CC08PM 145954740 Ki = 419.2 nM T53378 CNE86C 145954868 Ki = 6 nM T53378 C1LFA9 145954917 Ki = 5601 nM T53378 CMZ2Y0 145954932 Ki = 386.7 nM T53378 C6UGK8 145955158 Ki = 395.4 nM T53378 C0UG3K 145955383 Ki = 8302.6 nM T53378 CHTR07 145955486 Ki = 3.3 nM T53378 CS6GA9 145955537 Ki = 39.7 nM T53378 C27JZH 145955576 Ki = 369.5 nM T53378 CW90OF 145955720 Ki = 7.8 nM T53378 CB86QZ 145955914 Ki = 1350.2 nM T53378 CG7W8R 145955929 Ki = 2813.9 nM T53378 CDWF95 145955978 Ki = 1692.1 nM T53378 CDJV68 145956076 Ki = 2721.6 nM T53378 C5W1UM 145956081 Ki = 7228.7 nM T53378 CY1AD2 145956169 Ki = 1.7 nM T53378 CD3LK5 145956229 Ki = 173.5 nM T53378 C2KV9S 145956347 Ki = 1036.5 nM T53378 CGY39T 145956363 Ki = 326.2 nM T53378 CEL63H 145956491 Ki = 139 nM T53378 C4LH5W 145956563 Ki = 79.3 nM T53378 C7K2DA 145957040 Ki = 3643.4 nM T53378 CEF41D 145957103 Ki = 3510.9 nM T53378 CAMD59 145957136 Ki = 30.6 nM T53378 C94GRZ 145957236 Ki = 319.4 nM T53378 CED18K 145957307 Ki = 1180.7 nM T53378 C17FUI 145957430 Ki = 320.9 nM T53378 CN5TM2 145957461 Ki = 342.5 nM T53378 C4S7BR 145957546 Ki = 2887.8 nM T53378 CL28OB 145957582 Ki = 3837.7 nM T53378 CP4TF7 145957664 Ki = 156.1 nM T53378 C6HG7S 145957711 Ki = 2577.4 nM T53378 CE4O0N 145957959 Ki = 2.9 nM T53378 CXFV43 145958041 Ki = 211.4 nM T53378 CF07KV 145958447 Ki = 52.4 nM T53378 C5URQ2 145958565 Ki = 72.5 nM T53378 C0PRJ7 145958803 Ki = 4 nM T53378 C0F9NS 145958940 Ki = 2296 nM T53378 CUBA42 145958994 Ki = 918.5 nM T53378 CXVC18 145959110 Ki = 2299.7 nM T53378 CNP7C0 145959116 Ki = 581.3 nM T53378 C1HML4 145959374 Ki = 146 nM T53378 C0LC9M 145959407 Ki = 2296.5 nM T53378 CGK4O1 145959409 Ki = 839.2 nM T53378 CJMU23 145959635 Ki = 242.3 nM T53378 CPL41Z 145959905 Ki = 403.1 nM T53378 CGZ1K8 145959957 Ki = 435.2 nM T53378 CL0NM5 145960039 Ki = 2.3 nM T53378 CH2K1A 145960207 Ki = 795 nM T53378 C6JND4 145960287 Ki = 34.8 nM T53378 C89GHI 145960779 Ki = 371 nM T53378 CT6U2G 145961010 Ki = 62.2 nM T53378 CDA7G0 145962071 Ki = 133.4 nM T53378 C14OZY 145962693 Ki = 2.3 nM T53378 C5VI0K 145964063 Ki = 898.2 nM T53378 CGTA80 145964130 Ki = 7264 nM T53378 C9DE8Y 145964275 Ki = 734.4 nM T53378 C4C9IE 145964340 Ki = 59.9 nM T53378 CK21BE 145964400 Ki = 5483 nM T53378 CAPU84 145964558 Ki = 92.8 nM T53378 C6FE1K 145964671 Ki = 6760 nM T53378 CTC21S 145964779 Ki = 908.7 nM T53378 C3F4IS 145965133 Ki = 4290.5 nM T53378 C6RZT2 145965743 Ki = 3040.7 nM T53378 CINP09 145966173 Ki = 4305.8 nM T53378 C2G8VU 145966250 Ki = 7557 nM T53378 C5X7FM 145966343 Ki = 2244.6 nM T53378 CCDI76 145966475 Ki = 63.7 nM T53378 CQ64RX 145966558 Ki = 811 nM T53378 CJ4D0R 145967030 Ki = 354.7 nM T53378 C7SUX3 145967040 Ki = 672.8 nM T53378 C7HZ6V 145967049 Ki = 3256.1 nM T53378 CP8Q9U 145967308 Ki = 2864.4 nM T53378 CFY3M6 145968026 Ki = 5423 nM T53378 CDYR51 145968242 Ki = 8023 nM T53378 C10PQH 145968245 Ki = 731.2 nM T53378 CKME70 145968701 Ki = 73.4 nM T53378 CX4D2R 145969379 Ki = 295.9 nM T53378 C9R4VB 145971458 Ki = 389.3 nM T53378 CZ71HS 145971486 Ki = 82.3 nM T53378 C73WMA 145971736 Ki = 80.2 nM T53378 C9P6UE 145971793 Ki = 235 nM T53378 C6DQK4 145972104 Ki = 2693 nM T53378 CO4V1G 145972192 Ki = 19 nM T53378 CYMF38 145972316 Ki = 301.3 nM T53378 CP9H1U 145972366 Ki = 4712.2 nM T53378 CD42QZ 145972397 Ki = 49.1 nM T53378 CZ2LP7 145972551 Ki = 2986.4 nM T53378 COJ6K4 145972603 Ki = 3682.3 nM T53378 CFXW14 145972912 Ki = 75.4 nM T53378 CF5KR4 145972986 Ki = 8136 nM T53378 C65ZVF 145973004 Ki = 2526.6 nM T53378 CN20BQ 145973308 Ki = 2897.3 nM T53378 C1I8GK 145973355 Ki = 1974.3 nM T53378 C9MZS1 145973465 Ki = 5996 nM T53378 C7Y3WO 145973882 Ki = 268.8 nM T53378 C2C1KE 145973952 Ki = 3299.6 nM T53378 CJ15WQ 145974101 Ki = 9.5 nM T53378 C7ZRI0 145974266 Ki > 10000 nM T53378 CX5U8J 145974401 Ki = 77.2 nM T53378 C2MF3Y 145974672 Ki = 928.9 nM T53378 C1QZ7F 145974710 Ki = 6857 nM T53378 CG5SL1 145974949 Ki = 765.9 nM T53378 CVPA83 145974992 Ki = 902.1 nM T53378 CDU4M5 145975077 Ki = 77.7 nM T53378 C3I2WU 145975151 Ki = 8654 nM T53378 C5U8RK 145975281 Ki = 395.5 nM T53378 C1VJD3 145975355 Ki = 4751 nM T53378 CBL8Y4 145975424 Ki = 7737 nM T53378 CT16KB 145975591 Ki = 1409 nM T53378 CZVK21 145975933 Ki = 7298 nM T53378 CQ08AT 145976207 Ki = 3.6 nM T53378 CI9C6U 145976539 Ki = 3053 nM T53378 CZ7QU1 145976656 Ki = 765.9 nM T53378 C2BIZ4 145976658 Ki = 2634 nM T53378 CHI26Q 145976735 Ki = 3877 nM T53378 CZWC63 145977536 Ki = 1598 nM T53378 CH3IC0 145977574 Ki > 10000 nM T53378 CUEB47 145977814 Ki = 519.1 nM T53378 C81JIQ 145977869 Ki = 8627 nM T53378 CL7GH8 145977904 Ki = 1972.7 nM T53378 C69UQY 145978025 Ki = 522.6 nM T53378 C5QSK0 145978140 Ki = 101.9 nM T53378 CYG69V 145978605 Ki = 3005 nM T53378 CYWK54 145978673 Ki = 2804 nM T53378 C2D1TO 145978690 Ki = 441.9 nM T53378 CA32BT 145978780 Ki = 219.8 nM T53378 CFUC92 145979600 Ki = 392.4 nM T53378 C8YA0B 145979831 Ki = 3098 nM T53378 C5S9JX 145979949 Ki = 203.9 nM T53378 CD1IJ2 145980204 Ki = 751 nM T53378 CE3DP8 145980765 Ki = 216.5 nM T53378 C15PEL 145982039 Ki = 6353 nM T53378 C2O8PK 145982576 Ki = 79.2 nM T53378 CK8MY4 145982622 Ki = 229.4 nM T53378 CX6Y5G 145982786 Ki = 295.4 nM T53378 C7M0HW 145982836 Ki = 44.3 nM T53378 C34LIQ 145982969 Ki = 59.8 nM T53378 CH3EF7 145983056 Ki = 66.2 nM T53378 CN7G5J 145983107 Ki = 736.1 nM T53378 C90VNX 145983131 Ki = 648.7 nM T53378 CWUJ59 145983568 Ki = 84 nM T53378 CF26VG 145983797 Ki = 884.9 nM T53378 C5SLN9 145983850 Ki = 49.5 nM T53378 CI52KO 145983856 Ki = 229.5 nM T53378 C8PM9Y 145984067 Ki = 35.7 nM T53378 CA6I9T 145984095 Ki = 53 nM T53378 CEA52W 145984222 Ki = 36.6 nM T53378 CO9P3M 145984354 Ki = 628.2 nM T53378 C49ALP 145984517 Ki = 277.9 nM T53378 CLDZ58 145984801 Ki = 44.8 nM T53378 C05FCU 145984802 Ki = 169.2 nM T53378 C7N6ZB 145984855 Ki = 85.7 nM T53378 C4FBS2 145985005 Ki = 152.9 nM T53378 CZ8NA9 145985353 Ki = 88.3 nM T53378 C8Y1UT 145985534 Ki = 36.2 nM T53378 CF16KP 145985651 Ki = 9386 nM T53378 CJEG52 145985679 Ki = 2506.7 nM T53378 CN1WK4 145985761 Ki = 478.4 nM T53378 CIT98E 145985912 Ki = 836.1 nM T53378 C8VIF2 145985922 Ki = 569.7 nM T53378 CX0YW6 145985969 Ki = 272.5 nM T53378 C3E0RD 145986123 Ki = 1954.2 nM T53378 CF7CH8 145986297 Ki = 49.9 nM T53378 C9UBE8 145987408 Ki = 120.8 nM T53378 C65QOW 145987697 Ki = 652.3 nM T53378 C6RMF1 145987996 Ki = 853.9 nM T53378 C89RFU 145988368 Ki = 5155 nM T53378 CXA6F3 145988572 Ki = 941.1 nM T53378 CYJ79A 145989992 Ki = 2695 nM T53378 C9F8TL 145992666 Ki = 384.7 nM T53378 C7OZD6 145993265 Ki = 359.5 nM T53378 CS40WA 145993323 Ki = 873.1 nM T53378 CK3YT9 145993866 Ki = 6860 nM T53378 C48CZD 146160385 Ki = 220.1 nM T53378 C6FD2N 147348395 Ki = 452.4 nM T53378 C06MEW 155510831 Ki = 4.5 nM T53378 C1PG9M 155511036 Ki = 1.7 nM T53378 CN6DW9 155511075 Ki = 1644 nM T53378 C2PXC3 155511133 Ki = 1716.5 nM T53378 C03BJU 155511800 Ki = 39200 nM T53378 CJA94W 155512108 Ki = 192.1 nM T53378 C1ZPW3 155512418 Ki = 37.8 nM T53378 CQC04P 155512706 Ki = 41.9 nM T53378 C21CAW 155513169 Ki = 1004.7 nM T53378 CX2UJ9 155514131 Ki = 11000 nM T53378 CZ5W1M 155514230 Ki > 10000 nM T53378 CM5J3L 155514471 Ki = 1.2 nM T53378 CDM78Q 155514660 Ki = 21.9 nM T53378 CCQB03 155515285 Ki = 915.5 nM T53378 CZN16J 155516304 Ki = 68.7 nM T53378 COP4Q6 155516517 Ki = 2356 nM T53378 C7IR3P 155516553 Ki = 4500 nM T53378 C2E0ZF 155517026 Ki = 433.2 nM T53378 CAG9L4 155517430 Ki = 3555 nM T53378 CHA2R1 155517933 Ki = 21.1 nM T53378 C1VNX3 155518220 Ki = 2619 nM T53378 CEH62Y 155518447 Ki = 0.61 nM T53378 CP7UI1 155518510 Ki = 1196 nM T53378 CM7DQ6 155518807 Ki = 63.8 nM T53378 C8MYG2 155519248 Ki = 1322 nM T53378 CO6D1Y 155519288 Ki = 1389 nM T53378 CC47MV 155519432 Ki = 433.8 nM T53378 CO4V0B 155519627 Ki = 957.5 nM T53378 CIV68R 155520019 Ki = 424.6 nM T53378 CP49HE 155520274 Ki > 10000 nM T53378 C5JCL6 155520507 Ki = 59.7 nM T53378 CE8QY5 155520792 Ki = 111.9 nM T53378 C4LPA1 155520806 Ki > 10000 nM T53378 C2J1YG 155521041 Ki = 643.9 nM T53378 CCGT71 155521462 Ki = 608.5 nM T53378 CF7HE1 155521700 Ki = 2.1 nM T53378 CZ7WI8 155521830 Ki = 222.5 nM T53378 C6AWP0 155522679 Ki = 2.4 nM T53378 CA9F2I 155523252 Ki = 419.8 nM T53378 C3HGK6 155523328 Ki = 859.9 nM T53378 C3MX7F 155523857 Ki = 43.1 nM T53378 CS21YC 155524712 Ki = 80.5 nM T53378 C70ZPH 155524915 Ki = 810.4 nM T53378 CPL80N 155525961 Ki = 76.1 nM T53378 CA02GS 155526086 Ki = 1.8 nM T53378 CAMY18 155527145 Ki = 145 nM T53378 CDE96Y 155527673 Ki = 6415.6 nM T53378 CDN05K 155527975 Ki = 204.3 nM T53378 CLF2V0 155528496 Ki = 8695.3 nM T53378 C38SKR 155528605 Ki = 7364 nM T53378 C2LF1H 155528761 Ki = 6.5 nM T53378 C52QUD 155529352 Ki = 838.9 nM T53378 C8DN2F 155529373 Ki = 0.66 nM T53378 C2JV7R 155529885 Ki = 5239 nM T53378 CG3J0Q 155529984 Ki = 9719.5 nM T53378 CW07EO 155530326 Ki = 45.8 nM T53378 CKO2V5 155530358 Ki = 1984 nM T53378 CIGQ50 155530440 Ki = 974.4 nM T53378 CTJ3I7 155530506 Ki > 10000 nM T53378 CLMZ93 155531382 Ki = 307.6 nM T53378 CYBD02 155531537 Ki = 58300 nM T53378 C0BNY7 155533528 Ki = 1.8 nM T53378 CTKI39 155533898 Ki = 2958.4 nM T53378 C78ZFI 155534074 Ki = 42.1 nM T53378 CT5NG1 155534179 Ki = 9724 nM T53378 CS0FK9 155534753 Ki = 607.9 nM T53378 CVU5P6 155535355 Ki = 96.6 nM T53378 CKR07J 155535598 Ki > 10000 nM T53378 CFYA23 155535780 Ki = 31.3 nM T53378 C0EDQ2 155536876 Ki = 713.3 nM T53378 CZ0T6A 155537018 Ki = 2674 nM T53378 COP2R4 155537042 Ki = 25.1 nM T53378 C6T7BQ 155537167 Ki = 25600 nM T53378 CYM0A3 155538069 Ki = 1.5 nM T53378 C5RV9W 155538073 Ki = 443.6 nM T53378 COX74J 155538083 Ki = 0.9 nM T53378 C9AP8F 155538224 Ki = 1516 nM T53378 CB8C4X 155538289 Ki = 4300 nM T53378 C9K2TL 155539730 Ki > 10000 nM T53378 CS1G5V 155539783 Ki = 4456 nM T53378 CS1UR7 155539868 Ki = 958 nM T53378 CSAD81 155540401 Ki = 371.1 nM T53378 CZ8FJ3 155540422 Ki = 4.7 nM T53378 C7Z6FC 155541724 Ki = 62.2 nM T53378 C8RV6T 155541805 Ki = 1613 nM T53378 CW96ES 155541807 Ki = 746.5 nM T53378 C4MW9Q 155541811 Ki = 778.4 nM T53378 CX20DK 155541945 Ki = 19800 nM T53378 CW61DF 155542555 Ki = 7380 nM T53378 CT9GZ2 155542660 Ki > 10000 nM T53378 CDK2W5 155542691 Ki = 0.39 nM T53378 CY3BO6 155542934 Ki = 2004.1 nM T53378 C75TVG 155542954 Ki = 183.2 nM T53378 CN2SJ7 155543228 Ki = 542.9 nM T53378 C19DJA 155543271 Ki > 10000 nM T53378 CI2T8N 155544664 Ki = 71.7 nM T53378 C95IJM 155545916 Ki = 3444 nM T53378 CSW62L 155546892 Ki > 100000 nM T53378 C83ZIS 155547526 Ki = 259.2 nM T53378 C73YLV 155547628 Ki = 18.1 nM T53378 C61MSB 155547730 Ki = 6.8 nM T53378 CQG5F9 155548326 Ki = 2633 nM T53378 CDC0F4 155548911 Ki = 4.8 nM T53378 CU1NE7 155549031 Ki = 7186 nM T53378 CA25QH 155549266 Ki = 885.6 nM T53378 C8NS5F 155549723 Ki = 35600 nM T53378 C3YN0W 155550099 Ki = 4611.6 nM T53378 C4O6TN 155550616 Ki = 76.9 nM T53378 C6XPV0 155550626 Ki = 521.3 nM T53378 CTE04H 155551088 Ki = 29700 nM T53378 CPRC19 155551316 Ki = 256.6 nM T53378 C4S0JZ 155551334 Ki = 4164 nM T53378 COC4Z9 155551784 Ki = 292.4 nM T53378 C3AN2K 155551935 Ki = 12200 nM T53378 CG9PN8 155552113 Ki = 0.65 nM T53378 C7E3UF 155552316 Ki = 32200 nM T53378 CW8S7L 155552594 Ki = 84.8 nM T53378 CBQ42J 155552773 Ki = 1900 nM T53378 C1R7CJ 155553759 Ki = 9.6 nM T53378 CMEP40 155554179 Ki = 120.1 nM T53378 CM4I0O 155554763 Ki = 3100 nM T53378 CZU9Y7 155554800 Ki = 387 nM T53378 C5YA7C 155555084 Ki = 0.59 nM T53378 CA7UK2 155555803 Ki = 225.5 nM T53378 CWB82E 155555878 Ki = 6491 nM T53378 C9I0QN 155556147 Ki = 42.3 nM T53378 CGZ58Y 155556761 Ki = 61.7 nM T53378 C87GRH 155557329 Ki = 302.8 nM T53378 CRK5I0 155557428 Ki = 16200 nM T53378 C40MOH 155557452 Ki = 382.8 nM T53378 CZ7C0S 155558990 Ki = 127.7 nM T53378 C3Y7WJ 155560101 Ki = 23600 nM T53378 C3FG8W 155561198 Ki = 1400 nM T53378 CU03LF 155561751 Ki = 4338.4 nM T53378 CU1JV7 155561839 Ki = 4665.8 nM T53378 CXE2R9 155561928 Ki = 96 nM T53378 C6KD7C 155563215 Ki > 10000 nM T53378 CP85AZ 155563623 Ki = 0.31 nM T53378 CQ40DU 155563908 Ki = 6276 nM T53378 C07GFY 155564664 Ki = 0.22 nM T53378 C0E4QV 155565149 Ki = 906.5 nM T53378 CJ7I6Z 155565419 Ki = 360.3 nM T53378 CD6Z0B 155566206 Ki = 39.1 nM T53378 CJQP47 155566378 Ki = 0.52 nM T53378 CI8U3W 155566755 Ki = 0.89 nM T53378 C9DOG1 155567981 Ki = 4306.5 nM T53378 CZP30I 155567991 Ki = 1908.8 nM T53378 CG82MB 155568274 Ki = 1808.6 nM T53378 C94QKZ 155568447 Ki > 10000 nM T53378 CH5VU6 155568899 Ki = 6390 nM T53378 C83MGT 155569151 Ki = 1 nM T53378 CAUR85 155569555 Ki = 4800 nM T53378 C1A7IN 155569676 Ki = 1477 nM T53378 D00BMI 25154729 Ki = 8910 nM T53378 D00CIW 15295 Ki = 5400 nM T53378 D00IUB 13019 Ki = 634000 nM T53378 D00RNZ 910172 Ki = 5800 nM T53378 D00XJA 711717 Ki > 500000 nM T53378 D00YEF 148885 Ki = 91.2 nM T53378 D01BUB 94952 Ki = 426000 nM T53378 D01STY 9861037 Ki = 125 nM T53378 D01UYI 5281607 Ki = 537.75 nM T53378 D02DBP 5054 Ki = 570000 nM T53378 D02QGI 273 Ki = 52 nM T53378 D03NBX 637308 Ki = 44000 nM T53378 D03ZMQ 323 Ki = 6800 nM T53378 D04CVC 4687472 Ki = 180 nM T53378 D04NSN 169682 Ki = 348.8 nM T53378 D04PSK 44571848 Ki = 8300 nM T53378 D05KTE 6224 Ki = 99 nM T53378 D05QUG 45485279 Ki = 37400 nM T53378 D05TLB 11117301 Ki = 79.9 nM T53378 D05WQF 637540 Ki = 62300 nM T53378 D05XZM 10081162 Ki = 560 nM T53378 D06ALC 6441498 Ki = 101.2 nM T53378 D06DYP 234562 Ki = 31700 nM T53378 D06JVR 44571849 Ki = 5540 nM T53378 D07MTM 403 Ki = 743000 nM T53378 D07PZQ 68841 Ki = 4260000 nM T53378 D07QJJ 289 Ki = 10900 nM T53378 D07TAJ 914298 Ki = 7200 nM T53378 D07YDN 5281654 Ki = 212.9 nM T53378 D08AIJ 440735 Ki = 72.8 nM T53378 D08BFU 5282102 Ki = 5591.2 nM T53378 D09JPC 16402 Ki = 450 nM T53378 D09QHC 7370 Ki = 1120 nM T53378 D09UQM 97463 Ki = 890 nM T53378 D09WSJ 19772348 Ki = 67.6 nM T53378 D09WVV 8111 Ki = 116000 nM T53378 D0A0YX 5143 Ki = 7920 nM T53378 D0A1CM 5281855 Ki = 9080 nM T53378 D0A6HS 6852129 Ki = 17 nM T53378 D0AU0M 637542 Ki = 9600 nM T53378 D0C7LR 313 Ki = 90000 nM T53378 D0CM3O 446142 Ki = 5360000 nM T53378 D0D4OV 20043772 Ki = 84.1 nM T53378 D0D5XC 101753 Ki = 9900 nM T53378 D0D6UR 12394434 Ki = 27900 nM T53378 D0E3VJ 25154731 Ki = 7580 nM T53378 D0EJ9B 66827 Ki = 880 nM T53378 D0G3BI 25090 Ki = 8500 nM T53378 D0G3TK 5280863 Ki > 10000 nM T53378 D0G6OW 23675285 Ki = 74500 nM T53378 D0GQ9A 44593649 Ki = 870 nM T53378 D0H0PQ 278 Ki = 9900 nM T53378 D0H3NS 10752 Ki = 9700 nM T53378 D0IB3K 5320686 Ki = 5468.7 nM T53378 D0J2AE 7377 Ki = 2200 nM T53378 D0L2GD 60167587 Ki = 9800 nM T53378 D0L5TZ 20195365 Ki = 7700 nM T53378 D0LJ5P 44457221 Ki = 1356.8 nM T53378 D0LU4S 156219 Ki = 61200 nM T53378 D0M3PO 69561 Ki = 4830 nM T53378 D0M6RM 7365 Ki = 870 nM T53378 D0N1AW 45485270 Ki = 15000 nM T53378 D0NN3Q 78105 Ki = 3200 nM T53378 D0O1QT 93505 Ki = 19 nM T53378 D0OI1H 72894 Ki = 1310 nM T53378 D0OT5L 1631814 Ki > 500000 nM T53378 D0P6AM 3526523 Ki = 66 nM T53378 D0Q7DJ 10742 Ki = 10600 nM T53378 D0R7QY 127676 Ki = 1040 nM T53378 D0RB0D 44268050 Ki = 26800 nM T53378 D0S4NO 25154730 Ki = 8640 nM T53378 D0S9YX 5280373 Ki = 7078.5 nM T53378 D0SY2M 5281708 Ki = 718.7 nM T53378 D0T2VH 44571846 Ki = 8400 nM T53378 D0T6VB 521293 Ki = 30000 nM T53378 D0U4BB 10748 Ki = 8300 nM T53378 D0V9EN 689043 Ki = 10100 nM T53378 D0VD7H 84724 Ki = 540 nM T53378 D0X5HL 15107 Ki = 58 nM T53378 D0X6IE 4422372 Ki = 84 nM T53378 D0Y3TZ 370 Ki = 9800 nM T53378 D0Y7HG 5281616 Ki = 568.3 nM T53378 D0YU8J 1502014 Ki = 320 nM T53378 D0Z1HY 67136 Ki = 160 nM T61792 D00BCP 2727 IC50 = 133000 nM T61792 D00BLL 9849808 IC50 = 133000 nM T61792 D00DKK 5282379 IC50 = 133000 nM T61792 D00FGO 460612 IC50 = 133000 nM T61792 D00IBN 54676228 IC50 = 133000 nM T61792 D00KVO 2082 IC50 = 133000 nM T61792 D00MIN 657298 IC50 = 133000 nM T61792 D00NKB 5546 IC50 = 133000 nM T61792 D00WAM 3647 IC50 = 133000 nM T61792 D00WUF 5486971 IC50 = 133000 nM T61792 D00XUN 23894 IC50 = 133000 nM T61792 D00YZA 5453 IC50 = 133000 nM T61792 D00YZD 54726191 IC50 > 90000 nM T61792 D01AJY 2284 IC50 = 133000 nM T61792 D01AZG 5073 IC50 = 133000 nM T61792 D01DBQ 452548 IC50 = 133000 nM T61792 D01GBY 124087 IC50 = 133000 nM T61792 D01KKQ 135400182 IC50 = 133000 nM T61792 D01MDT 5487 IC50 = 133000 nM T61792 D01MUR 68844 IC50 = 133000 nM T61792 D01OXI 2578 IC50 = 133000 nM T61792 D01STB 5362129 IC50 = 133000 nM T61792 D01UTL 2995 IC50 = 133000 nM T61792 D01UXC 2249 IC50 = 133000 nM T61792 D01XNB 4594 IC50 = 133000 nM T61792 D01XYJ 35370 IC50 = 133000 nM T61792 D01ZII 2726 IC50 = 133000 nM T61792 D01ZSO 4235 IC50 = 133000 nM T61792 D02DGU 444795 IC50 = 133000 nM T61792 D02DPA 2756 IC50 = 133000 nM T61792 D02FEM 5284447 IC50 = 133000 nM T61792 D02HED 4748 IC50 = 133000 nM T61792 D02LCR 5467 IC50 = 133000 nM T61792 D02NTO 5510 IC50 = 133000 nM T61792 D02STN 132971 IC50 = 133000 nM T61792 D02TLO 3690 IC50 = 133000 nM T61792 D02YIZ 12560 IC50 = 133000 nM T61792 D03CQE 5379 IC50 = 133000 nM T61792 D03DDR 3034034 IC50 = 133000 nM T61792 D03ELL 2159 IC50 = 133000 nM T61792 D03HJK 447043 IC50 = 133000 nM T61792 D03JSJ 446596 IC50 = 133000 nM T61792 D03KOZ 1549120 IC50 = 84400 nM T61792 D03KQF 4011 IC50 = 133000 nM T61792 D03KZM 216237 IC50 = 133000 nM T61792 D03NHW 4583 IC50 = 133000 nM T61792 D03QWT 73303 IC50 = 133000 nM T61792 D03RTS 2662 IC50 = 133000 nM T61792 D03TVW 54120 IC50 = 133000 nM T61792 D03TYI 9433 IC50 = 133000 nM T61792 D03VPC 2754 IC50 = 133000 nM T61792 D03XOC 656583 IC50 = 133000 nM T61792 D03YLZ 27200 IC50 = 133000 nM T61792 D04AAW 60613 IC50 = 133000 nM T61792 D04ASH 657180 IC50 = 80200 nM T61792 D04EGX 54746 IC50 = 133000 nM T61792 D04FBR 5281078 IC50 = 133000 nM T61792 D04ITO 6436173 IC50 = 15400 nM T61792 D04JCN 47811 IC50 = 133000 nM T61792 D04JEE 4946 IC50 = 133000 nM T61792 D04JPJ 3950 IC50 = 133000 nM T61792 D04KYY 135401907 IC50 = 133000 nM T61792 D04MSM 2554 IC50 = 133000 nM T61792 D04NXQ 51081 IC50 = 133000 nM T61792 D04OSE 4485 IC50 = 133000 nM T61792 D04RGA 5282415 IC50 = 133000 nM T61792 D04VMT 5253 IC50 = 133000 nM T61792 D04WFD 4543 IC50 = 133000 nM T61792 D04XGT 31593 IC50 = 133000 nM T61792 D04YMH 151166 IC50 = 133000 nM T61792 D04ZTY 444020 IC50 = 133000 nM T61792 D05AFX 4450 IC50 = 133000 nM T61792 D05ARP 135398740 IC50 = 133000 nM T61792 D05DVP 5717 IC50 = 58800 nM T61792 D05EAM 4735 IC50 = 133000 nM T61792 D05FTJ 4044 IC50 = 133000 nM T61792 D05GJW 20279 IC50 = 133000 nM T61792 D05HPI 16134395 IC50 = 29100 nM T61792 D05HSC 6000 IC50 = 133000 nM T61792 D05LEO 3385 IC50 = 133000 nM T61792 D05LKP 5215 IC50 = 133000 nM T61792 D05MFA 135398741 IC50 = 133000 nM T61792 D05MQK 110635 IC50 = 133000 nM T61792 D05OFX 219078 IC50 = 133000 nM T61792 D05UVD 33624 IC50 = 133000 nM T61792 D05VIL 5284594 IC50 = 133000 nM T61792 D05VLS 5090 IC50 = 133000 nM T61792 D05ZGQ 5281070 IC50 = 133000 nM T61792 D05ZIK 4205 IC50 = 133000 nM T61792 D06ABF 3957 IC50 = 133000 nM T61792 D06BEP 2712 IC50 = 133000 nM T61792 D06CTE 57469 IC50 = 133000 nM T61792 D06FDR 135398739 IC50 = 133000 nM T61792 D06GAM 3357 IC50 = 133000 nM T61792 D06GDY 43815 IC50 = 133000 nM T61792 D06JPB 5280793 IC50 = 133000 nM T61792 D06NXY 5991 IC50 = 133000 nM T61792 D06OIV 5505 IC50 = 133000 nM T61792 D06OMK 445643 IC50 = 40300 nM T61792 D06OVY 5362065 IC50 = 89400 nM T61792 D06PSS 5311309 IC50 = 133000 nM T61792 D06TNL 3278 IC50 = 3850 nM T61792 D06UDG 60846 IC50 = 133000 nM T61792 D06WTZ 53232 IC50 = 133000 nM T61792 D06XAE 1712095 IC50 = 133000 nM T61792 D06XMU 6013 IC50 = 133000 nM T61792 D06YYD 9578005 IC50 = 133000 nM T61792 D06ZII 969472 IC50 = 133000 nM T61792 D06ZUK 3696 IC50 = 133000 nM T61792 D07ABV 468595 IC50 = 133000 nM T61792 D07BCT 36294 IC50 = 133000 nM T61792 D07CWD 3657 IC50 = 133000 nM T61792 D07DJQ 10219 IC50 = 133000 nM T61792 D07HGR 5362119 IC50 = 133000 nM T61792 D07HVY 64139 IC50 = 133000 nM T61792 D07IEF 2391 IC50 = 133000 nM T61792 D07IPB 454216 IC50 = 64000 nM T61792 D07JGT 4421 IC50 = 133000 nM T61792 D07KSG 2733526 IC50 = 133000 nM T61792 D07POC 176870 IC50 = 10000 nM T61792 D07QCE 2265 IC50 = 133000 nM T61792 D07SUG 2478 IC50 = 133000 nM T61792 D07TQV 60825 IC50 = 133000 nM T61792 D07UYO 441401 IC50 = 133000 nM T61792 D07VDZ 5284627 IC50 = 133000 nM T61792 D07VLY 31703 IC50 = 133000 nM T61792 D07WEP 3019 IC50 = 133000 nM T61792 D07XGR 3339 IC50 = 133000 nM T61792 D07XSN 6253 IC50 = 133000 nM T61792 D08EBN 41684 IC50 = 133000 nM T61792 D08HVR 6047 IC50 = 133000 nM T61792 D08IWD 57363 IC50 = 133000 nM T61792 D08JIV 2162 IC50 = 133000 nM T61792 D08PIQ 6741 IC50 = 133000 nM T61792 D08QIP 4887 IC50 = 133000 nM T61792 D08ROP 3899 IC50 = 133000 nM T61792 D08USJ 4456 IC50 = 133000 nM T61792 D08VRO 3822 IC50 = 133000 nM T61792 D08VXL 5353788 IC50 = 133000 nM T61792 D08VYV 4168 IC50 = 133000 nM T61792 D08ZEB 2733 IC50 = 133000 nM T61792 D09CZA 5282226 IC50 = 133000 nM T61792 D09DHY 6167 IC50 = 133000 nM T61792 D09DWL 5719 IC50 = 133000 nM T61792 D09EGZ 2719 IC50 = 133000 nM T61792 D09HNR 3002190 IC50 = 133000 nM T61792 D09HVL 16129704 IC50 = 133000 nM T61792 D09IOI 2170 IC50 = 133000 nM T61792 D09IPV 28417 IC50 = 133000 nM T61792 D09JUG 60490 IC50 = 133000 nM T61792 D09LNI 3365 IC50 = 133000 nM T61792 D09LWS 150311 IC50 = 133000 nM T61792 D09MGR 123619 IC50 = 133000 nM T61792 D09NIA 2732 IC50 = 133000 nM T61792 D09QEI 4740 IC50 = 133000 nM T61792 D09TBD 5344 IC50 = 133000 nM T61792 D09WEJ 2446 IC50 = 133000 nM T61792 D09XQF 3767 IC50 = 133000 nM T61792 D09XZB 123631 IC50 = 133000 nM T61792 D0A0OO 65016 IC50 = 133000 nM T61792 D0A2ZX 4173 IC50 = 133000 nM T61792 D0A5SE 134018 IC50 = 133000 nM T61792 D0A9YA 6918296 IC50 = 133000 nM T61792 D0AA2D 2378 IC50 = 133000 nM T61792 D0AD5C 41774 IC50 = 133000 nM T61792 D0AN7B 896 IC50 = 133000 nM T61792 D0AO5H 5578 IC50 = 133000 nM T61792 D0AP9T 53025 IC50 = 133000 nM T61792 D0AV3G 3151 IC50 = 133000 nM T61792 D0AZ3C 5291 IC50 = 133000 nM T61792 D0B1IP 5282375 IC50 = 133000 nM T61792 D0B2UZ 4917 IC50 = 133000 nM T61792 D0B3HD 2519 IC50 = 133000 nM T61792 D0B5MP 135398513 IC50 = 133000 nM T61792 D0B6TW 135403647 IC50 = 133000 nM T61792 D0B7EB 36462 IC50 = 133000 nM T61792 D0B7NG 2725 IC50 = 133000 nM T61792 D0B8UJ 3011155 IC50 = 133000 nM T61792 D0BA9U 13109 IC50 = 133000 nM T61792 D0BM5G 5381 IC50 = 133000 nM T61792 D0BP9C 193962 IC50 = 7800 nM T61792 D0C3YQ 23662354 IC50 = 133000 nM T61792 D0C4RB 36314 IC50 = 133000 nM T61792 D0C6NM 5311221 IC50 = 133000 nM T61792 D0C8EU 5394 IC50 = 133000 nM T61792 D0CL9S 159269 IC50 = 133000 nM T61792 D0CT9C 2907 IC50 = 133000 nM T61792 D0CW1P 9782 IC50 = 133000 nM T61792 D0D0BE 28061 IC50 = 133000 nM T61792 D0D0ZD 441314 IC50 = 133000 nM T61792 D0D1AL 3559 IC50 = 133000 nM T61792 D0D1SG 5755 IC50 = 133000 nM T61792 D0D2VS 60198 IC50 = 133000 nM T61792 D0D4JO 6917864 IC50 = 133000 nM T61792 D0D5GD 3373 IC50 = 133000 nM T61792 D0D5GG 4723 IC50 = 133000 nM T61792 D0D7KC 5488548 IC50 = 133000 nM T61792 D0D7LA 4091 IC50 = 133000 nM T61792 D0D8XY 5311010 IC50 = 133000 nM T61792 D0DJ1B 156391 IC50 = 133000 nM T61792 D0E0SW 53708 IC50 = 133000 nM T61792 D0E1SW 1986 IC50 = 133000 nM T61792 D0E1XL 5284583 IC50 = 133000 nM T61792 D0E6OC 5282230 IC50 = 133000 nM T61792 D0E6XR 3062316 IC50 = 133000 nM T61792 D0E6YQ 1935 IC50 = 133000 nM T61792 D0E7PQ 5311 IC50 = 133000 nM T61792 D0EG1I 9926791 IC50 = 133000 nM T61792 D0ES1Q 6918289 IC50 = 17600 nM T61792 D0F2PO 4828 IC50 = 133000 nM T61792 D0F6EO 33613 IC50 = 133000 nM T61792 D0F7CS 6758 IC50 = 133000 nM T61792 D0F8RA 2153 IC50 = 133000 nM T61792 D0F9GE 3108 IC50 = 133000 nM T61792 D0FM2P 82153 IC50 = 133000 nM T61792 D0G3DL 135398735 IC50 = 53000 nM T61792 D0G4OD 54686904 IC50 = 133000 nM T61792 D0G5AG 104762 IC50 = 133000 nM T61792 D0G5UB 2161 IC50 = 133000 nM T61792 D0G8NN 119570 IC50 = 133000 nM T61792 D0G9IU 135403821 IC50 = 16300 nM T61792 D0G9YH 2179 IC50 = 133000 nM T61792 D0GU4K 135413536 IC50 = 133000 nM T61792 D0GY5Z 2244 IC50 = 133000 nM T61792 D0H0KB 5070 IC50 = 133000 nM T61792 D0H0ND 54454 IC50 = 133000 nM T61792 D0H3HM 60795 IC50 = 133000 nM T61792 D0H3WI 37542 IC50 = 133000 nM T61792 D0H6QU 6005 IC50 = 133000 nM T61792 D0H8FH 3702 IC50 = 133000 nM T61792 D0I0EG 44093 IC50 = 133000 nM T61792 D0I2MK 4171 IC50 = 133000 nM T61792 D0I4DQ 5280723 IC50 = 133000 nM T61792 D0I6IB 54677971 IC50 = 133000 nM T61792 D0IT2G 5743 IC50 = 133000 nM T61792 D0IT2X 2581 IC50 = 133000 nM T61792 D0J1MI 4030 IC50 = 133000 nM T61792 D0J1VY 5281081 IC50 = 133000 nM T61792 D0J2KV 4932 IC50 = 133000 nM T61792 D0J2MJ 26758 IC50 = 133000 nM T61792 D0J4JM 5770 IC50 = 68400 nM T61792 D0J5DC 2796 IC50 = 133000 nM T61792 D0JC9N 60164 IC50 = 133000 nM T61792 D0JO7Y 104741 IC50 = 133000 nM T61792 D0JY3V 107751 IC50 = 133000 nM T61792 D0K0OZ 5702160 IC50 = 133000 nM T61792 D0K0VO 5639 IC50 = 133000 nM T61792 D0K3MC 3947 IC50 = 133000 nM T61792 D0K3QS 6442177 IC50 = 11300 nM T61792 D0K5CB 2083 IC50 = 133000 nM T61792 D0K6GZ 60464 IC50 = 133000 nM T61792 D0K7HU 6918155 IC50 = 133000 nM T61792 D0K7WK 4595 IC50 = 133000 nM T61792 D0K8KX 5280343 IC50 = 133000 nM T61792 D0KG3R 9875401 IC50 = 133000 nM T61792 D0KR2J 135398508 IC50 = 133000 nM T61792 D0L3DK 6918537 IC50 = 133000 nM T61792 D0L5RW 65015 IC50 = 133000 nM T61792 D0L5WM 2157 IC50 = 133000 nM T61792 D0L6DA 119607 IC50 = 133000 nM T61792 D0L7FM 4911 IC50 = 133000 nM T61792 D0L9ZR 4891 IC50 = 133000 nM T61792 D0M2MR 3475 IC50 = 133000 nM T61792 D0M3QP 441207 IC50 = 133000 nM T61792 D0M4YC 3114 IC50 = 133000 nM T61792 D0M5JI 9560989 IC50 = 133000 nM T61792 D0M6DO 2145 IC50 = 133000 nM T61792 D0M8RC 5403 IC50 = 133000 nM T61792 D0M8VE 71360 IC50 = 133000 nM T61792 D0M9BW 68911 IC50 = 133000 nM T61792 D0M9DC 4614 IC50 = 133000 nM T61792 D0MA9N 2955 IC50 = 133000 nM T61792 D0ML1F 60871 IC50 = 133000 nM T61792 D0N0RU 82146 IC50 = 133000 nM T61792 D0N0TZ 60606 IC50 = 133000 nM T61792 D0N1FS 26248 IC50 = 133000 nM T61792 D0N3VR 71616 IC50 = 133000 nM T61792 D0N4OW 644077 IC50 = 133000 nM T61792 D0N5HJ 5462501 IC50 = 133000 nM T61792 D0N5YA 65981 IC50 = 72300 nM T61792 D0N6RF 65999 IC50 = 133000 nM T61792 D0NG7O 60857 IC50 = 133000 nM T61792 D0NJ3V 4680 IC50 = 133000 nM T61792 D0NR6S 3002977 IC50 = 133000 nM T61792 D0NS6H 3152 IC50 = 133000 nM T61792 D0NW3X 71329 IC50 = 133000 nM T61792 D0O1WX 2764 IC50 = 133000 nM T61792 D0O2EM 4463 IC50 = 133000 nM T61792 D0O2SR 47528 IC50 = 133000 nM T61792 D0O3OS 104850 IC50 = 133000 nM T61792 D0O4SE 5479 IC50 = 133000 nM T61792 D0O5FY 441130 IC50 = 133000 nM T61792 D0O5WP 148124 IC50 = 133000 nM T61792 D0OB1J 39186 IC50 = 133000 nM T61792 D0OT0O 44561 IC50 = 133000 nM T61792 D0P1UX 5656 IC50 = 133000 nM T61792 D0P7JZ 34359 IC50 = 133000 nM T61792 D0P9RF 5401 IC50 = 133000 nM T61792 D0PQ3G 3440 IC50 = 133000 nM T61792 D0PW7C 51039 IC50 = 133000 nM T61792 D0Q2PE 4539 IC50 = 133000 nM T61792 D0Q2XF 5311027 IC50 = 133000 nM T61792 D0Q3YO 1547484 IC50 = 133000 nM T61792 D0Q4SD 443872 IC50 = 133000 nM T61792 D0Q4XQ 3291 IC50 = 133000 nM T61792 D0Q4YK 4843 IC50 = 133000 nM T61792 D0Q5NX 216326 IC50 = 133000 nM T61792 D0Q5UQ 214348 IC50 = 133000 nM T61792 D0Q6NZ 5281034 IC50 = 133000 nM T61792 D0Q8ZX 2337 IC50 = 133000 nM T61792 D0QL3P 34312 IC50 = 133000 nM T61792 D0R0BX 6604200 IC50 = 133000 nM T61792 D0R0FE 2520 IC50 = 133000 nM T61792 D0R1RS 3715 IC50 = 235000 nM T61792 D0R1WR 4919 IC50 = 133000 nM T61792 D0R2KJ 18381 IC50 = 133000 nM T61792 D0R3FP 6398764 IC50 = 133000 nM T61792 D0R3QY 5665 IC50 = 133000 nM T61792 D0R5RR 119182 IC50 = 133000 nM T61792 D0R8ER 3229 IC50 = 133000 nM T61792 D0R9OH 5329 IC50 = 133000 nM T61792 D0R9VR 9651 IC50 = 133000 nM T61792 D0S1NZ 5310993 IC50 = 133000 nM T61792 D0S3WH 68827 IC50 = 133000 nM T61792 D0S4BR 1349907 IC50 = 133000 nM T61792 D0S5CU 4499 IC50 = 133000 nM T61792 D0S5UH 2794 IC50 = 10400 nM T61792 D0S5WG 3366 IC50 = 133000 nM T61792 D0S9MC 2789 IC50 = 133000 nM T61792 D0S9SD 60877 IC50 = 133000 nM T61792 D0SH3I 387447 IC50 = 133000 nM T61792 D0SV8E 126941 IC50 = 133000 nM T61792 D0T0KA 4474 IC50 = 133000 nM T61792 D0T1LK 4908 IC50 = 133000 nM T61792 D0T2PL 5280453 IC50 = 133000 nM T61792 D0T2XU 4927 IC50 = 133000 nM T61792 D0T5WK 4506 IC50 = 133000 nM T61792 D0T7US 5281037 IC50 = 57900 nM T61792 D0T8GD 89594 IC50 = 133000 nM T61792 D0T9DT 2140 IC50 = 133000 nM T61792 D0T9TJ 3034010 IC50 = 133000 nM T61792 D0TR5X 3386 IC50 = 133000 nM T61792 D0U0KW 208902 IC50 = 133000 nM T61792 D0U2JP 4369359 IC50 = 133000 nM T61792 D0U4UQ 3639 IC50 = 133000 nM T61792 D0U5GB 92727 IC50 = 133000 nM T61792 D0U5QK 1983 IC50 = 133000 nM T61792 D0U5RT 4909 IC50 = 133000 nM T61792 D0U5SI 4913 IC50 = 133000 nM T61792 D0U8UV 10660 IC50 = 133000 nM T61792 D0UF6M 9568512 IC50 = 133000 nM T61792 D0UL2L 54690031 IC50 = 133000 nM T61792 D0UM7O 3821 IC50 = 133000 nM T61792 D0V4QS 135398745 IC50 = 133000 nM T61792 D0V7CF 5362440 IC50 = 133000 nM T61792 D0V8QT 2708 IC50 = 133000 nM T61792 D0V9BD 2375 IC50 = 133000 nM T61792 D0VM2L 68740 IC50 = 133000 nM T61792 D0VT8P 3324 IC50 = 133000 nM T61792 D0W0BF 2187 IC50 = 133000 nM T61792 D0W9LX 2585 IC50 = 133000 nM T61792 D0WI3T 441243 IC50 = 133000 nM T61792 D0WN0U 3333 IC50 = 133000 nM T61792 D0WS1X 6915944 IC50 = 133000 nM T61792 D0X0RI 4178 IC50 = 133000 nM T61792 D0X3FX 5284596 IC50 = 133000 nM T61792 D0X4RN 3676 IC50 = 133000 nM T61792 D0X5SD 3117 IC50 = 133000 nM T61792 D0X5XU 451668 IC50 = 133000 nM T61792 D0X6GN 444025 IC50 = 133000 nM T61792 D0X7DE 4449 IC50 = 133000 nM T61792 D0X7KZ 6918182 IC50 = 133000 nM T61792 D0X7XG 3000226 IC50 = 133000 nM T61792 D0X9RG 5361092 IC50 = 133000 nM T61792 D0X9ZC 47965 IC50 = 133000 nM T61792 D0XF8W 1046 IC50 = 133000 nM T61792 D0Y0SW 3397 IC50 = 133000 nM T61792 D0Y2CJ 4201 IC50 = 133000 nM T61792 D0Y3MO 37768 IC50 = 133000 nM T61792 D0Y5DO 2771 IC50 = 133000 nM T61792 D0Y5UG 2160 IC50 = 133000 nM T61792 D0Y7EM 3332 IC50 = 133000 nM T61792 D0Y7IU 5281004 IC50 = 133000 nM T61792 D0Y7ZU 135398738 IC50 = 133000 nM T61792 D0Y9LL 42884 IC50 = 133000 nM T61792 D0YV1Q 6032 IC50 = 133000 nM T61792 D0Z1RV 135398737 IC50 = 133000 nM T61792 D0Z1ZM 84029 IC50 = 133000 nM T61792 D0Z3DY 2333 IC50 = 41600 nM T61792 D0Z4EI 55245 IC50 = 133000 nM T61792 D0Z4SB 3478 IC50 = 133000 nM T61792 D0Z4UN 6509979 IC50 = 133000 nM T61792 D0Z5BC 5634 IC50 = 133000 nM T61792 D0Z6UC 5358 IC50 = 133000 nM T61792 D0Z7KE 3784 IC50 = 133000 nM T61792 D0Z8EX 18283 IC50 = 133000 nM T61792 D0Z9QR 24066 IC50 = 133000 nM T61792 D0ZB7K 5735 IC50 = 133000 nM T61792 D0ZS8P 2801 IC50 = 133000 nM T61792 D0ZU9R 392622 IC50 = 133000 nM T61792 D00TIG 6917964 IC50 = 133000 nM T61792 D02HTD 25167947 IC50 = 12000 nM T61792 D08YWK 6436 IC50 = 133000 nM T61792 D09YDM 24360 IC50 = 133000 nM T61792 D0CE0O 11513676 IC50 = 18000 nM T61792 D0E3TC 44259 IC50 = 133000 nM T61792 D0G7UX 5284373 IC50 = 13600 nM T61792 D0Q9CY 9915743 IC50 = 133000 nM T61792 D0SD9V 53276 IC50 = 133000 nM T61792 D0TO2R 30751 IC50 = 133000 nM T61792 D0V1WQ 24857286 IC50 = 2410 nM T61792 D0VG0D 11977753 IC50 = 133000 nM T61792 D0Y1FO 472335 IC50 = 60500 nM T61792 D01PIL 54477 IC50 = 133000 nM T61792 D01VAB 2119 IC50 = 133000 nM T61792 D02LHR 33625 IC50 = 133000 nM T61792 D03JPH 54677972 IC50 = 133000 nM T61792 D04BQR 4342 IC50 = 133000 nM T61792 D05RUM 15387 IC50 = 133000 nM T61792 D06ABW 2788 IC50 = 133000 nM T61792 D07GTB 16760063 IC50 = 20700 nM T61792 D07XPE 8249 IC50 = 133000 nM T61792 D08SOF 5405 IC50 = 133000 nM T61792 D0C0JT 4495 IC50 = 133000 nM T61792 D0D1LG 11995990 IC50 = 59000 nM T61792 D0G9ZW 54676478 IC50 = 133000 nM T61792 D0J9GD 64715 IC50 = 133000 nM T61792 D0O2IE 4754 IC50 = 133000 nM T61792 D0OS6O 60149 IC50 = 133000 nM T61792 D0P1JI 312145 IC50 = 46100 nM T61792 D0S6QR 214350 IC50 = 133000 nM T61792 D0Y2HR 2247 IC50 = 133000 nM T61792 D0Y4FL 6915744 IC50 = 133000 nM T61792 D0Y8UB 82148 IC50 = 133000 nM T61792 C85KQB 2202 IC50 = 133000 nM T61792 CI74WY 2450 IC50 = 133000 nM T61792 CPJ0C2 2747 IC50 = 133000 nM T61792 C36WOC 2800 IC50 = 133000 nM T61792 C7CT6M 2804 IC50 = 133000 nM T61792 CJ0B9F 3158 IC50 = 133000 nM T61792 C0H8GR 3191 IC50 = 133000 nM T61792 CEXU05 3383 IC50 = 133000 nM T61792 COSX53 3519 IC50 = 133000 nM T61792 CO2Y3R 3698 IC50 = 133000 nM T61792 C4ZJT8 3730 IC50 = 133000 nM T61792 CY4WG9 3793 IC50 = 133000 nM T61792 C9LCD8 3823 IC50 = 133000 nM T61792 C2KJI7 3883 IC50 = 133000 nM T61792 C12UDR 4411 IC50 = 133000 nM T61792 C8VXJ6 4888 IC50 = 133000 nM T61792 C93BJO 5039 IC50 = 133000 nM T61792 C48GPY 5475 IC50 = 133000 nM T61792 C1EYR7 5497 IC50 = 133000 nM T61792 C2U1WA 6216 IC50 = 133000 nM T61792 C59UQE 6279 IC50 = 133000 nM T61792 CC09DB 9703 IC50 = 133000 nM T61792 CO1I7C 11080 IC50 = 133000 nM T61792 CMU2P6 11683 IC50 = 133000 nM T61792 C2J7BV 12947 IC50 = 133000 nM T61792 CVJ2X3 14051 IC50 = 133000 nM T61792 C6RG5E 21233 IC50 = 133000 nM T61792 CJ3OL7 25590 IC50 = 133000 nM T61792 CK21BO 27350 IC50 = 133000 nM T61792 C4VU9Z 31098 IC50 = 133000 nM T61792 CUJ6W7 35455 IC50 = 133000 nM T61792 CZA2C6 39764 IC50 = 133000 nM T61792 CFX82C 47320 IC50 = 133000 nM T61792 C6E5CD 48229 IC50 = 133000 nM T61792 CE8LA7 49659 IC50 = 133000 nM T61792 CU86VK 54459 IC50 = 133000 nM T61792 C7ZUJ4 54840 IC50 = 133000 nM T61792 CC10UB 56801 IC50 = 133000 nM T61792 CQSF39 57004 IC50 = 133000 nM T61792 CH8GS0 60749 IC50 = 133000 nM T61792 CYQ4S7 60822 IC50 = 133000 nM T61792 CHZJ65 60834 IC50 = 133000 nM T61792 C2GKD5 62884 IC50 = 133000 nM T61792 CA9S6G 62978 IC50 = 133000 nM T61792 C7SO5H 63021 IC50 = 133000 nM T61792 CP8F7B 64143 IC50 = 133000 nM T61792 CD9TC8 64737 IC50 = 133000 nM T61792 C7WUM6 65335 IC50 = 133000 nM T61792 COZ10X 65348 IC50 = 133000 nM T61792 CS7L6J 65957 IC50 = 133000 nM T61792 C7AV1G 68553 IC50 = 133000 nM T61792 C73LEV 71399 IC50 = 133000 nM T61792 C6A4VW 71651 IC50 = 133000 nM T61792 C2F1OT 77997 IC50 = 133000 nM T61792 C1W8YJ 78000 IC50 = 133000 nM T61792 C6NLX4 84003 IC50 = 133000 nM T61792 CVP7G8 101526 IC50 = 133000 nM T61792 C90TYQ 130313 IC50 = 133000 nM T61792 CAR7Y4 146571 IC50 = 133000 nM T61792 C3WVZ6 154068 IC50 = 133000 nM T61792 C4J5ZF 185617 IC50 = 75000 nM T61792 CI7BE6 219025 IC50 = 133000 nM T61792 CA6ID2 241903 IC50 = 133000 nM T61792 CV80FO 249332 IC50 = 133000 nM T61792 C0VN3D 288216 IC50 = 133000 nM T61792 CLD6J9 441074 IC50 = 133000 nM T61792 CY7HM4 441313 IC50 = 133000 nM T61792 CDU0B1 441351 IC50 = 133000 nM T61792 CVX0K8 443866 IC50 = 133000 nM T61792 C40YBS 444036 IC50 = 133000 nM T61792 C35HJB 656684 IC50 = 133000 nM T61792 CGIY90 688272 IC50 = 133000 nM T61792 CBM17N 3000706 IC50 = 133000 nM T61792 C4BR7C 3005572 IC50 = 133000 nM T61792 CWQI02 3033817 IC50 = 133000 nM T61792 CH86TV 3033968 IC50 = 133000 nM T61792 C2XP0H 3052775 IC50 = 133000 nM T61792 CONV41 4022878 IC50 = 133000 nM T61792 C4SL8Q 5281025 IC50 = 133000 nM T61792 C9QDT1 5281067 IC50 = 133000 nM T61792 CNI9X4 5281888 IC50 = 133000 nM T61792 C4X7RJ 5282408 IC50 = 133000 nM T61792 C10CPM 5282455 IC50 = 133000 nM T61792 CBLX43 5282481 IC50 = 133000 nM T61792 CB4P2S 5289394 IC50 = 133000 nM T61792 CUA96S 5388961 IC50 = 133000 nM T61792 C5DV8U 5702270 IC50 = 133000 nM T61792 C4GST2 6321416 IC50 = 133000 nM T61792 CC9WJ2 6433334 IC50 = 133000 nM T61792 CQR03B 6526396 IC50 = 133000 nM T61792 C0P8LZ 6602611 IC50 = 133000 nM T61792 CPK20Z 6917733 IC50 = 133000 nM T61792 C9FQ0W 6918092 IC50 = 133000 nM T61792 C9P2HT 9556529 IC50 = 133000 nM T61792 CEO67P 9588170 IC50 = 133000 nM T61792 C5W7MS 9833407 IC50 = 133000 nM T61792 CJL94H 9839243 IC50 = 133000 nM T61792 C7QK8R 9847786 IC50 = 133000 nM T61792 CIWP56 9886273 IC50 = 133000 nM T61792 C5NH4J 9912089 IC50 = 133000 nM T61792 C45JHO 9933004 IC50 = 133000 nM T61792 CIV15Q 10113978 IC50 = 133000 nM T61792 CY73KI 10322450 IC50 > 50000 nM T61792 C8BL9W 10695961 IC50 = 133000 nM T61792 C63EXW 11463807 EC50 = 145000 nM T61792 CVG4M1 11679357 IC50 = 133000 nM T61792 C67LTO 11995989 IC50 = 100000 nM T61792 C7K8VQ 11996131 EC50 = 71000 nM T61792 CUG2Q8 11996283 IC50 = 200000 nM T61792 C47ZJY 11996857 IC50 = 50000 nM T61792 CZ6PB5 12001375 IC50 = 133000 nM T61792 CCLY36 12004215 IC50 = 133000 nM T61792 CT0DU8 13633111 IC50 > 200000 nM T61792 CO9ES2 13633119 IC50 = 21500 nM T61792 C9N5YG 14720269 IC50 = 133000 nM T61792 CGL5Q2 16051965 IC50 = 133000 nM T61792 CA3JL7 16052011 IC50 = 133000 nM T61792 C7WI4H 16204922 IC50 = 133000 nM T61792 CLHO84 16759173 IC50 = 133000 nM T61792 C71VGO 16760285 IC50 = 133000 nM T61792 CUZE40 18004026 IC50 = 133000 nM T61792 C28AYI 18530292 IC50 = 64200 nM T61792 C0REQ9 20055509 IC50 = 133000 nM T61792 CQ31BP 23623618 IC50 = 133000 nM T61792 CFE9R6 23666879 IC50 = 133000 nM T61792 CH59NC 23667631 IC50 = 133000 nM T61792 CWB0H2 23674512 IC50 = 56200 nM T61792 CFLN18 23675322 IC50 = 133000 nM T61792 CD01LT 23685176 IC50 = 133000 nM T61792 C9YI0H 23716436 IC50 = 133000 nM T61792 C3N4GQ 25078429 IC50 = 133000 nM T61792 CM80XH 25222999 IC50 > 20000 nM T61792 C26ZQR 25223001 IC50 > 50000 nM T61792 CKY89F 25223106 IC50 > 50000 nM T61792 C03FQV 25223201 IC50 > 20000 nM T61792 C8S6UH 25223298 IC50 > 20000 nM T61792 C24GQB 25223515 EC50 = 140000 nM T61792 CW7ZK4 44181971 IC50 = 133000 nM T61792 CG18FA 44563898 IC50 < 150 nM T61792 CUA6N3 46783232 IC50 = 133000 nM T61792 C9SCG4 49800073 IC50 = 133000 nM T61792 CRV3P5 54685920 IC50 = 133000 nM T61792 CGK7Y9 54685925 IC50 = 133000 nM T61792 CQ6C4E 56972143 IC50 = 133000 nM T61792 CM5T1V 57393422 IC50 = 133000 nM T61792 CI5Y1T 69003097 IC50 = 12200 nM T61792 CTO71V 72734347 IC50 = 133000 nM T61792 CRZ62F 73355036 IC50 = 36800 nM T61792 CFDV48 86288862 IC50 = 14400 nM T61792 COVK20 90142631 IC50 = 140000 nM T61792 C5BPR6 90676904 IC50 = 9000 nM T61792 CUO89W 90676905 IC50 = 11100 nM T61792 CV57FY 90676982 IC50 = 10600 nM T61792 CP4N5J 90676984 IC50 = 10500 nM T61792 C7ZX1M 90676986 IC50 = 17500 nM T61792 CQP6J4 90676989 IC50 = 11400 nM T61792 CPT43K 90676990 IC50 = 4500 nM T61792 C6JYI5 90676991 IC50 = 6300 nM T61792 C0GJE9 90676992 IC50 = 4800 nM T61792 C30OFR 90676993 IC50 = 13900 nM T61792 C3YZ5E 134139366 IC50 = 4500 nM T61792 CH34YB 134140743 IC50 = 15800 nM T61792 CQGK07 134143225 IC50 = 17800 nM T61792 CG0VJ9 134146560 IC50 = 8200 nM T61792 CKA90D 134147852 IC50 = 15400 nM T61792 CDF35J 134150848 IC50 = 7300 nM T61792 CVTI13 134154345 IC50 = 4100 nM T61792 C41TDB 135413523 IC50 = 133000 nM T61792 CDN1S3 135413539 IC50 = 133000 nM T61792 CG8C4T 135415564 IC50 = 49800 nM T61792 C27TMO 137648451 IC50 = 133000 nM T61792 CHPC06 137654606 IC50 = 133000 nM T61792 C67IKZ 145948937 IC50 = 133000 nM T61792 C7GK3H 145990715 IC50 > 100000 nM T61792 C9RLJ3 3661 IC50 = 133000 nM T61792 D00RFY 5281612 IC50 > 50000 nM T61792 D01FGM 5280666 IC50 > 50000 nM T61792 D01OIK 155774 IC50 = 133000 nM T61792 D03IRR 2206 IC50 = 133000 nM T61792 D07GXY 4850 IC50 = 133000 nM T61792 D08CNS 3748 IC50 = 133000 nM T61792 D09XCX 5694 IC50 = 133000 nM T61792 D0F4QX 5601 IC50 = 133000 nM T61792 D0F5LH 4634 IC50 = 133000 nM T61792 D0J6JT 1355 IC50 = 133000 nM T61792 D0L9PX 5943 IC50 = 133000 nM T61792 D0T3PW 5281672 IC50 = 22000 nM T61792 D0T5RO 16129706 IC50 = 133000 nM T07279 D00IFR 58423153 Ki = 0.16 nM T07279 D03HUX 49792852 IC50 > 10000 nM T07279 D03LWG 53235510 IC50 > 10000 nM T07279 D07EHV 44814409 Ki = 0.018 nM T07279 D09JEJ 24748573 IC50 = 186 nM T07279 D0E3TC 44259 IC50 = 21.7 nM T07279 D0W3LI 153999 IC50 > 20000 nM T07279 D04VSB 68356857 IC50 = 12 nM T07279 D06OKX 68356855 IC50 = 18 nM T07279 D08JUU 68327881 IC50 = 41 nM T07279 D0J6HN 46179018 Ki = 0.002 nM T07279 D0OS2I 59226518 Ki = 0.002 nM T07279 D0P9UF 51002052 Ki = 5 nM T07279 D0T3ME 156422 IC50 > 30000 nM T07279 CG5XY6 1201120 IC50 = 100 nM T07279 C5PDS4 1206018 IC50 = 300 nM T07279 CQ7PL4 1235170 IC50 > 20000 nM T07279 C2REL7 1239884 IC50 = 2300 nM T07279 C2JSX4 1241442 IC50 = 4700 nM T07279 CFX90H 1243769 IC50 = 40 nM T07279 C8I0WK 1361334 Ki = 100 nM T07279 CM3CE2 1379638 IC50 > 100000 nM T07279 CIB51E 1379720 IC50 = 400 nM T07279 CEW8K1 1379922 IC50 = 160 nM T07279 COTN75 1382447 IC50 = 200 nM T07279 CWJS81 1539584 IC50 = 2500 nM T07279 CB8K9W 1641790 IC50 = 90 nM T07279 C03SAD 1641793 IC50 = 100 nM T07279 CH4TI3 2243909 IC50 = 100 nM T07279 CGK6Q2 3157072 IC50 > 100000 nM T07279 C9DL5A 5878179 IC50 = 43000 nM T07279 CH1R8P 5985287 IC50 = 4400 nM T07279 C1GZ5L 6006914 IC50 = 80 nM T07279 CAH19P 6026872 IC50 = 40 nM T07279 C4J5VQ 6076476 IC50 = 20 nM T07279 C7GP2B 9965755 IC50 = 900 nM T07279 C3K7CB 10236138 IC50 = 13500 nM T07279 CBOP58 11293798 Ki > 10000 nM T07279 C26BZX 11362471 Ki > 10000 nM T07279 CWXB93 11397177 Ki > 10000 nM T07279 CTG83F 11539329 Ki > 1400 nM T07279 CACS26 11561968 Ki > 2000 nM T07279 CMIL86 11590363 Ki > 1400 nM T07279 C9T6SC 11640926 Ki > 1400 nM T07279 CU0E8O 11690457 Ki > 2000 nM T07279 CDFI41 13365773 IC50 = 7100 nM T07279 CFPW41 16007116 Ki > 1400 nM T07279 COPQ34 16043794 Ki = 250 nM T07279 C38FDZ 16760660 IC50 = 110 nM T07279 CBG4X2 20784957 Ki = 15000 nM T07279 CG0NS1 24737654 IC50 = 12 nM T07279 CQNP54 24764449 IC50 = 25000 nM T07279 C4Z9CN 24769780 IC50 > 25000 nM T07279 CP1WR0 24795070 IC50 = 362 nM T07279 C5TJ4H 24811473 IC50 = 265 nM T07279 C2N9HS 24811474 IC50 = 25 nM T07279 CLCU03 24811585 IC50 = 22 nM T07279 C2DHS8 24811587 IC50 = 94 nM T07279 CX08QH 24811590 IC50 = 140 nM T07279 CPKH12 24811592 IC50 = 27 nM T07279 CF16OG 24811687 IC50 = 370 nM T07279 C0K7NB 24811691 IC50 = 480 nM T07279 C5RH1W 24811692 IC50 = 310 nM T07279 C50PCT 24811792 IC50 = 1020 nM T07279 C5R1ZV 24811793 IC50 = 17 nM T07279 CY8X0J 24811794 IC50 = 40 nM T07279 CVQI42 24811797 IC50 = 10 nM T07279 CNU5W2 24811798 IC50 = 150 nM T07279 CN8MC2 24811902 IC50 = 200 nM T07279 C39CPS 24811905 IC50 = 880 nM T07279 C3SLC1 24811908 IC50 = 1700 nM T07279 C1X2RU 24812007 IC50 = 3300 nM T07279 C73WEX 24812008 IC50 = 46 nM T07279 CNX6L4 24812011 IC50 > 8000 nM T07279 CZ7P6C 24853967 IC50 = 161000 nM T07279 C4D2QE 24894053 Ki = 0.004 nM T07279 CX1HL8 25032704 Ki = 43.5 nM T07279 C0B7RT 25057409 IC50 > 10000 nM T07279 CS2P3O 25185171 IC50 = 2200 nM T07279 CLG79A 25185172 IC50 > 100000 nM T07279 C90BFN 25185173 IC50 = 100000 nM T07279 CMI7T4 25185174 IC50 > 100000 nM T07279 CLH4S6 25185175 IC50 > 100000 nM T07279 C3QF7Z 25185441 IC50 > 100000 nM T07279 C0R4PY 25185442 IC50 > 100000 nM T07279 C19MTD 25185443 IC50 > 100000 nM T07279 CO6L0V 25185444 IC50 > 100000 nM T07279 CDN2V4 25189319 IC50 = 1500 nM T07279 C2DSU0 25189321 IC50 = 42000 nM T07279 C46UKS 25189322 IC50 = 500 nM T07279 CIY3A2 25190453 Ki = 174 nM T07279 CN0YI4 25190454 Ki = 62.8 nM T07279 C0YXD8 25190455 Ki = 165 nM T07279 CC10AL 25190456 Ki = 558 nM T07279 CHP23Y 25190458 Ki > 1424 nM T07279 CIWV65 25190459 Ki > 1424 nM T07279 C1KY2L 25190460 Ki > 1424 nM T07279 C19AOI 25190461 Ki > 1424 nM T07279 C8V0PL 25190462 Ki > 1424 nM T07279 CP7T1I 25263224 IC50 = 1200 nM T07279 C3BU1V 25263225 IC50 = 1400 nM T07279 C1P2LT 25263227 IC50 = 2200 nM T07279 CL85GI 39005031 Ki > 12500 nM T07279 CUQE83 44187007 IC50 = 7 nM T07279 C9V3XY 44199470 Ki = 0.05 nM T07279 CU13JS 44217530 Ki < 3 nM T07279 CW96TZ 44217683 Ki = 6 nM T07279 CBW35D 44222957 IC50 = 18 nM T07279 C0LDV8 44222965 IC50 = 3 nM T07279 C3ZJ6S 44222969 IC50 = 12 nM T07279 CX4SQ0 44222970 IC50 = 12 nM T07279 CAG56N 44222977 IC50 = 20 nM T07279 CPJ3G8 44241505 IC50 = 510 nM T07279 CL3M2Q 44545852 IC50 = 25 nM T07279 CL4SE1 44573315 IC50 = 160 nM T07279 CWQ1Z6 44573316 IC50 > 8000 nM T07279 C01GEN 44581101 IC50 > 100000 nM T07279 CEQN62 44609163 IC50 = 5 nM T07279 C7G4FT 44609164 IC50 = 5 nM T07279 CH9FO5 44609165 IC50 < 3 nM T07279 CLPY85 44609168 IC50 < 4 nM T07279 CU0QT2 44609322 IC50 < 4 nM T07279 CQ06VN 44609327 IC50 < 3 nM T07279 CE9GN6 44609485 IC50 = 14 nM T07279 C4QC7B 44609634 IC50 = 250 nM T07279 C37RDC 45110412 IC50 = 2460 nM T07279 CV7S5L 45110413 IC50 = 980 nM T07279 CU3RF1 45139989 IC50 > 10000 nM T07279 CQGZ06 45139991 IC50 > 10000 nM T07279 CDS4J9 46178380 Ki < 3 nM T07279 CP0WY1 46178460 Ki = 23 nM T07279 C4S8MP 46179491 Ki = 4 nM T07279 CY3HW5 46224684 IC50 > 10000 nM T07279 C7ON5A 46233287 IC50 > 10000 nM T07279 CLS29B 46872626 IC50 > 10000 nM T07279 C2O8RZ 46886323 IC50 > 1000 nM T07279 C09RXA 46937301 IC50 = 131 nM T07279 C2HZ3M 49779260 IC50 = 41 nM T07279 CAZ1V8 49805556 IC50 = 43 nM T07279 CF91RS 49843531 IC50 > 10000 nM T07279 CVQ6P3 50915164 IC50 = 2 nM T07279 C68POW 50941395 IC50 = 94 nM T07279 CF3YB2 50941397 IC50 = 294 nM T07279 CX93HP 50942535 IC50 > 2500 nM T07279 C71RUL 50942628 IC50 > 2500 nM T07279 CZ8B9T 50942630 IC50 = 1250 nM T07279 CUG03K 51033838 IC50 = 4 nM T07279 C5NT2O 51036049 IC50 = 8 nM T07279 CK0MX5 51036250 IC50 = 28 nM T07279 C4RH7Z 51036450 IC50 = 2 nM T07279 C1RN8T 51036645 IC50 = 2 nM T07279 CO7MY6 51036646 IC50 = 9 nM T07279 CEG98T 51036856 IC50 = 25 nM T07279 C7B1JO 51037081 IC50 = 34 nM T07279 CDTC84 51037916 IC50 = 6 nM T07279 C4PI9Q 51351831 IC50 = 54 nM T07279 C3DTV5 53233133 IC50 = 190 nM T07279 C82IWE 53250611 IC50 = 13800 nM T07279 C0SWH5 53348216 IC50 > 40000 nM T07279 CNI7P9 53372541 IC50 = 230 nM T07279 C0IYG7 53372543 IC50 = 69 nM T07279 CA6H2P 53372668 IC50 = 1000 nM T07279 CY1I9B 53372669 IC50 = 218 nM T07279 COP26H 53372670 IC50 = 404 nM T07279 CFM7W8 53372672 IC50 = 752 nM T07279 C9GYZ3 53372790 IC50 = 29 nM T07279 C8NA4L 53384644 IC50 > 30000 nM T07279 C49DRM 53482602 Ki = 0.1 nM T07279 CS4Y9F 53482665 Ki = 8.1 nM T07279 CR9P7C 53482785 Ki = 5 nM T07279 C5IWB4 53482960 Ki = 2 nM T07279 C2AJ9L 54576042 IC50 = 390 nM T07279 CQFH98 54580157 IC50 = 11900 nM T07279 CR1UO2 54580158 IC50 = 100 nM T07279 CA43ED 54581151 IC50 = 5800 nM T07279 C3H9FS 54581152 IC50 = 590 nM T07279 C56PNV 54581153 IC50 = 21 nM T07279 CG4FR6 54581154 IC50 = 250 nM T07279 C75IDW 54581155 IC50 = 21100 nM T07279 C9IL8D 54581156 IC50 = 260 nM T07279 C3N8XT 54581186 IC50 = 6100 nM T07279 CVNC57 54582208 IC50 = 1300 nM T07279 C0TZ7R 54583142 IC50 = 150 nM T07279 C73GAJ 54583143 IC50 = 350 nM T07279 C1NLW0 54585070 IC50 = 330 nM T07279 CJO3M1 54585071 IC50 = 340 nM T07279 CN73GO 54585072 IC50 = 1300 nM T07279 CH6CE1 54586044 IC50 = 160 nM T07279 CF7B2S 54586045 IC50 = 1200 nM T07279 CYD87G 54586046 IC50 = 12500 nM T07279 CI9U5M 54586075 IC50 = 7000 nM T07279 CH03RW 54587027 IC50 = 2900 nM T07279 CL38AX 54587028 IC50 = 540 nM T07279 CWQ31J 54752779 IC50 = 83 nM T07279 CZ4CR6 54752780 IC50 = 61 nM T07279 C96CIG 54752781 IC50 = 81 nM T07279 C2FK8I 54752782 IC50 = 56 nM T07279 C1XS2J 54760383 IC50 > 10000 nM T07279 CM8JX1 56604907 IC50 = 25000 nM T07279 CC7T2A 56674921 IC50 = 70 nM T07279 CBOD63 56835089 IC50 > 30000 nM T07279 CN8YK1 56935642 IC50 = 21 nM T07279 CFKA67 57390288 IC50 = 15000 nM T07279 CYF74P 57390289 IC50 > 25000 nM T07279 C4Y3WA 57390290 IC50 = 20 nM T07279 CU3WM8 57390291 IC50 = 10 nM T07279 CGT82N 57390292 IC50 = 26 nM T07279 CO92HZ 57390346 IC50 = 10 nM T07279 CC3X4H 57390347 IC50 = 10 nM T07279 CS0Y1G 57392065 IC50 > 25000 nM T07279 C13ARH 57392066 IC50 > 25000 nM T07279 CAD9Q1 57392067 IC50 = 174 nM T07279 CD7R3C 57392125 IC50 = 8 nM T07279 CG5LM0 57392126 IC50 = 5 nM T07279 C53YDP 57392127 IC50 = 2 nM T07279 CZT5Q4 57392128 IC50 = 4 nM T07279 C1SGW3 57393817 IC50 > 25000 nM T07279 C34RIH 57393818 IC50 = 5000 nM T07279 C6I5MD 57393819 IC50 = 74 nM T07279 C6ZNF8 57393820 IC50 = 117 nM T07279 CT2IK5 57393821 IC50 = 55 nM T07279 C24ITU 57393822 IC50 = 10 nM T07279 C1K4BX 57393824 IC50 = 113 nM T07279 CYK23D 57393887 IC50 = 18 nM T07279 CHG95S 57393892 IC50 = 5 nM T07279 CA28OK 57393893 IC50 = 2 nM T07279 C6PN4T 57393894 IC50 = 4 nM T07279 CD6Y9Z 57395116 IC50 > 30000 nM T07279 C8W6IG 57395117 IC50 > 30000 nM T07279 C29ZPK 57395544 IC50 = 42 nM T07279 CWV27Q 57395545 IC50 = 650 nM T07279 CGJ67T 57395546 IC50 = 26 nM T07279 C04UWN 57395547 IC50 = 92 nM T07279 CQEL83 57395548 IC50 = 59 nM T07279 C82EYJ 57395549 IC50 = 44 nM T07279 CXN51F 57395611 IC50 = 894 nM T07279 CS4Q7E 57395612 IC50 > 2500 nM T07279 C42ESL 57395623 IC50 = 8 nM T07279 CL58MG 57395624 IC50 = 5 nM T07279 CSZ37K 57396179 IC50 > 25000 nM T07279 CE2YT1 57396291 IC50 = 2 nM T07279 CW4KG3 57396858 IC50 = 853 nM T07279 CG7S0D 57396882 IC50 > 30000 nM T07279 CIBU80 57397370 IC50 > 25000 nM T07279 CC6Q2N 57397371 IC50 = 26 nM T07279 CNC93S 57397372 IC50 = 6 nM T07279 C0F3LV 57397435 IC50 = 1 nM T07279 C70URD 57397436 IC50 = 12 nM T07279 C1UZP2 57397437 IC50 = 6 nM T07279 C1L4HY 57398127 IC50 = 350 nM T07279 CODG52 57398624 IC50 = 358 nM T07279 C0PNU8 57399041 IC50 = 20 nM T07279 C4CW2G 57400284 IC50 = 640 nM T07279 CC73VO 57400785 IC50 > 25000 nM T07279 CM7NS6 57400786 IC50 = 72 nM T07279 CX5MH0 57400787 IC50 = 122 nM T07279 CD47VK 57400788 IC50 = 158 nM T07279 CR29GW 57400789 IC50 = 8 nM T07279 C3G5BY 57400790 IC50 = 15 nM T07279 CAD5G6 57400791 IC50 = 31 nM T07279 C6QIJ2 57400845 IC50 > 2500 nM T07279 C9NJ0A 57400853 IC50 = 8 nM T07279 CM24WI 57400854 IC50 = 1 nM T07279 CJ4YR1 57400855 IC50 = 10 nM T07279 C36ZSI 57402544 IC50 = 7200 nM T07279 C6F9HJ 57402545 IC50 = 20000 nM T07279 CVBS23 57402546 IC50 = 13600 nM T07279 CG35HA 57402547 IC50 = 10 nM T07279 CW7I5C 57402548 IC50 = 16 nM T07279 C9GXO5 57402606 IC50 = 54 nM T07279 CA71NH 57403845 IC50 > 1000 nM T07279 C6JET5 58182164 Ki = 2.2 nM T07279 CPU40N 58189477 IC50 = 9 nM T07279 C2B4KD 58189484 IC50 = 68 nM T07279 CGML85 58189493 IC50 = 28 nM T07279 C4PI2X 58189496 IC50 = 6 nM T07279 CL85RA 58189505 IC50 = 14 nM T07279 CD96SU 58189506 IC50 = 17 nM T07279 C3J0BF 58189523 IC50 = 76 nM T07279 C3ZAY9 58189525 IC50 = 24 nM T07279 C1QM9E 58189526 IC50 = 7 nM T07279 CL5J0G 58189527 IC50 = 86 nM T07279 C6P8JQ 58189528 IC50 = 5 nM T07279 C3X1OD 58189540 IC50 = 121 nM T07279 CCJW98 58189542 IC50 = 12 nM T07279 C63GUR 58189549 IC50 = 52 nM T07279 CP12HS 58189553 IC50 = 17 nM T07279 CI8QG4 58189555 IC50 = 15 nM T07279 CP3YX7 58189559 IC50 = 4 nM T07279 CE96XT 58189563 IC50 = 12 nM T07279 CL3AQ9 58189570 IC50 = 6 nM T07279 CLB8X2 58189576 IC50 = 5 nM T07279 C37EVM 58189578 IC50 = 21 nM T07279 CO87KC 58189587 IC50 = 49 nM T07279 CL5R9Q 58189614 IC50 = 6 nM T07279 CJ9RY1 58189624 IC50 = 52 nM T07279 C8GU4K 58189625 IC50 = 22 nM T07279 CO06IF 58189629 IC50 = 15 nM T07279 C78RDU 58189641 IC50 = 10 nM T07279 CXT6Q2 58423155 IC50 = 180 nM T07279 C73BEA 58423187 IC50 = 15000 nM T07279 C3KL4R 58423251 IC50 = 82 nM T07279 CF0L6E 58423275 IC50 = 25 nM T07279 CY2I5D 58423319 IC50 = 79 nM T07279 CBY0I7 58423384 IC50 = 500 nM T07279 CRG4K0 58464982 Ki = 0.4 nM T07279 CLE79F 59190121 IC50 = 38 nM T07279 CW7F1B 59190170 IC50 = 445 nM T07279 CC3HF5 59190198 IC50 = 62 nM T07279 CEI9F1 59190242 IC50 = 109 nM T07279 C4T8QV 59190250 IC50 = 127 nM T07279 C7E3JK 59190306 IC50 = 5 nM T07279 C6H8IU 59226389 Ki = 5 nM T07279 CCU1I6 59455685 Ki = 29 nM T07279 C4KV1J 59587678 IC50 = 20 nM T07279 CGV9W1 59587708 IC50 = 30 nM T07279 C1MR8Q 60097495 IC50 > 1000 nM T07279 C4BRH3 62046501 Ki > 12500 nM T07279 CK6WO0 66552478 IC50 < 10000 nM T07279 C90ZFG 66597948 IC50 = 4090 nM T07279 CHO3M7 66597981 IC50 = 269 nM T07279 CYO8V7 66597989 IC50 = 8160 nM T07279 C7W2XF 66597997 IC50 = 228 nM T07279 C16DNF 66598062 IC50 = 732 nM T07279 C4RCD5 66598081 IC50 = 100 nM T07279 C38XNO 66598093 IC50 = 987 nM T07279 C52HRW 66598095 IC50 = 282 nM T07279 C82RIS 66598100 IC50 = 2070 nM T07279 CRDF75 66598125 IC50 = 6020 nM T07279 CF9T4M 66598126 IC50 = 506 nM T07279 C1ET4P 66598128 IC50 = 1491 nM T07279 C5D3TJ 66598153 IC50 = 525 nM T07279 CJFZ71 66598162 IC50 = 2040 nM T07279 CG7X8T 66598186 IC50 = 639 nM T07279 CF5R9E 66598190 IC50 = 1260 nM T07279 CBS45L 66615214 IC50 = 1020 nM T07279 C8LT0N 66615220 IC50 = 4660 nM T07279 CJ31XD 66615233 IC50 = 3620 nM T07279 CX8T5L 66772114 IC50 = 38 nM T07279 CV63UL 67240318 IC50 > 10000 nM T07279 C7FCH0 67959600 IC50 = 16 nM T07279 CB65ES 67959736 IC50 = 9 nM T07279 CTK1D8 67959952 IC50 = 58 nM T07279 CE54CI 67960005 IC50 = 3000 nM T07279 CY3AZ9 67960061 IC50 = 1.1 nM T07279 CV8O1G 67960139 IC50 = 70 nM T07279 CVFC41 67960161 IC50 = 33 nM T07279 CP2G8D 67960181 IC50 = 3 nM T07279 CR7DN8 68032650 IC50 = 22 nM T07279 CGO14Q 68161034 Ki = 35 nM T07279 C02UIN 68161275 Ki = 110 nM T07279 C4XZ5Q 68161316 Ki > 12500 nM T07279 CA0UR4 68161594 Ki = 50 nM T07279 CY0QN9 68161639 Ki = 2000 nM T07279 CD41ZA 68161763 Ki = 700 nM T07279 C0US3B 68161865 Ki = 120 nM T07279 C36FUI 68161871 Ki = 4 nM T07279 CYJQ86 68162030 Ki = 187 nM T07279 C6FEN2 68162062 Ki = 8 nM T07279 CJR94B 68162223 Ki = 317 nM T07279 CAD7C0 68162522 Ki = 27 nM T07279 C9GJN4 68162758 Ki = 680 nM T07279 C09NJI 68162802 Ki < 3 nM T07279 C57KXW 68162851 Ki = 158 nM T07279 C97XLW 68163204 Ki < 3 nM T07279 C1E3XF 68184638 Ki = 4 nM T07279 C3SFB2 68184734 Ki = 16 nM T07279 C9XD8R 68187352 Ki < 3 nM T07279 CH2FV7 68187375 Ki = 0.2 nM T07279 CN6A5W 68187418 Ki < 3 nM T07279 CYM62W 68187421 Ki = 70 nM T07279 CYR6N1 68187478 Ki < 1 nM T07279 C7YX8H 68187480 Ki < 3 nM T07279 CKD38R 68187493 Ki = 7 nM T07279 CU3L1D 68187495 Ki = 8 nM T07279 CY6CG5 68187593 Ki = 6 nM T07279 CUB29K 68187641 Ki = 12 nM T07279 C4VUW2 68328157 IC50 = 114 nM T07279 CA19JZ 68328195 IC50 = 28 nM T07279 CC5F2N 68328262 IC50 = 1010 nM T07279 CDP01I 68328283 IC50 = 22 nM T07279 CA1NW4 68328307 IC50 = 6 nM T07279 C2PK9C 68328329 IC50 = 59 nM T07279 CM5NV2 68328390 IC50 = 104 nM T07279 COQ2P8 68328395 IC50 = 25 nM T07279 CRT84L 68328588 IC50 = 21 nM T07279 CGP7B8 68328695 IC50 = 348 nM T07279 C67HDR 68328735 IC50 = 227 nM T07279 C7O9RP 68356711 IC50 = 2220 nM T07279 C7GRD4 68356716 IC50 = 10 nM T07279 CYP10F 68356783 IC50 = 977 nM T07279 CQ6VX1 68356838 IC50 = 37 nM T07279 CUKO28 68356850 IC50 = 192 nM T07279 C4JR8X 68356863 IC50 = 1630 nM T07279 CT8O2I 69042864 Ki = 0.006 nM T07279 CSD25R 69045198 Ki = 94 nM T07279 C5NL7W 69047229 Ki < 3 nM T07279 CXI31L 69047447 Ki = 1600 nM T07279 C6QXP3 69090096 Ki = 6 nM T07279 C7B1IP 69090444 Ki = 4 nM T07279 CBJF23 70692372 IC50 = 82 nM T07279 C3O8YB 70694431 IC50 = 225 nM T07279 CAMN71 70696496 IC50 = 217 nM T07279 C3GDX9 70696694 IC50 = 690 nM T07279 CH0B8N 70789756 IC50 > 30000 nM T07279 CMAT40 70981556 IC50 > 1000 nM T07279 C7DO2P 70981589 IC50 = 3.4 nM T07279 C0WC3B 70981821 IC50 = 3.1 nM T07279 C23ARZ 70982089 IC50 = 1.6 nM T07279 C0Y8PA 70982249 IC50 = 148 nM T07279 CNKX61 70982376 IC50 = 2.9 nM T07279 CH7J2X 70982568 IC50 = 0.094 nM T07279 CM4T3D 70983036 IC50 = 1.6 nM T07279 C97WBL 70983181 IC50 = 0.18 nM T07279 C61DAP 70983443 IC50 = 0.43 nM T07279 C9ASG6 70984064 IC50 = 0.5 nM T07279 CVT09B 71007225 IC50 = 30 nM T07279 C1BND0 71007226 IC50 = 3.2 nM T07279 C35VQT 71007233 IC50 = 2.6 nM T07279 C0O7XS 71007248 IC50 = 1.1 nM T07279 CFD27U 71007268 IC50 > 1000 nM T07279 CWK3P9 71007275 IC50 = 27 nM T07279 C17CSR 71007292 IC50 = 31 nM T07279 CT23JC 71007294 IC50 = 5.4 nM T07279 C5DA2P 71007297 IC50 = 35 nM T07279 C34ANW 71007298 IC50 = 0.29 nM T07279 CILG13 71007335 IC50 = 11 nM T07279 C2K6EB 71007339 IC50 = 6.4 nM T07279 CZ1TG7 71007340 IC50 = 0.79 nM T07279 CR1G6M 71007342 IC50 = 6.5 nM T07279 C0KEC3 71007349 IC50 = 12 nM T07279 CBF2N4 71007352 IC50 = 110 nM T07279 C0XZ4A 71007357 IC50 = 2.2 nM T07279 CO3C5Z 71007358 IC50 = 49 nM T07279 C2WF8G 71202406 IC50 > 10000 nM T07279 CCN94X 71227735 IC50 = 2005 nM T07279 C4IEN5 71253342 Ki = 0.2 nM T07279 C6VHC3 71253383 Ki = 0.088 nM T07279 C3EF9T 71253391 Ki = 0.253 nM T07279 CQI4F0 71253507 Ki = 17 nM T07279 C8NX5J 71253513 Ki = 6.2 nM T07279 C9I2AE 71253517 Ki = 1.1 nM T07279 CTR6B1 71253520 Ki = 35 nM T07279 CP4SE3 71253554 Ki = 0.5 nM T07279 CH9RZ3 71253640 Ki = 4 nM T07279 CIN75X 71253646 Ki = 70 nM T07279 CI4BD1 71253671 Ki = 0.473 nM T07279 CU1QK9 71253681 Ki = 0.145 nM T07279 CZ9DL0 71253684 Ki = 50 nM T07279 CZA1B4 71253727 Ki = 2.2 nM T07279 CDJ29S 71253734 Ki = 0.58 nM T07279 CX7Z3V 71253771 Ki = 0.2 nM T07279 CPLG04 71253796 Ki = 0.3 nM T07279 C8YOC3 71253802 Ki = 14 nM T07279 C6QV8R 71253835 Ki = 0.72 nM T07279 CQL89K 71253906 Ki = 0.43 nM T07279 C6YKF5 71253921 Ki = 48 nM T07279 CUBE27 71253945 Ki = 170 nM T07279 CP60UQ 71253958 Ki = 3 nM T07279 CWRX87 71254005 Ki = 26 nM T07279 CCNF28 71254040 Ki = 8300 nM T07279 CJTH24 71254053 Ki = 1100 nM T07279 CW8H0Y 71254055 Ki = 800 nM T07279 C1W5TL 71254066 Ki = 1.25 nM T07279 COM7L3 71254090 Ki = 0.11 nM T07279 CBST91 71254178 Ki = 0.049 nM T07279 C1HB5Q 71254188 Ki = 0.127 nM T07279 C4GTF2 71254199 Ki = 3 nM T07279 CB7Z5W 71254288 Ki = 3 nM T07279 CA8G2O 71254348 Ki = 5.4 nM T07279 C2CJI8 71254349 Ki = 33 nM T07279 C2HKV3 71262574 IC50 = 36 nM T07279 C6RA0F 71262581 IC50 = 56 nM T07279 C9QE2L 71262654 IC50 = 14 nM T07279 C2OA1S 71262676 IC50 = 150 nM T07279 CS3E8P 71262754 IC50 = 1 nM T07279 C90JDF 71262764 IC50 = 18 nM T07279 CP0GU5 71262790 IC50 = 360 nM T07279 CZ89GY 71262793 IC50 = 400 nM T07279 C5DXK1 71307955 Ki = 0.032 nM T07279 CKT60L 71455860 Ki > 1400 nM T07279 C8Y3VW 71465328 IC50 = 1.3 nM T07279 C0LI2T 71488479 IC50 = 4260 nM T07279 CE41DB 71488550 IC50 = 690 nM T07279 CJR9V5 71488552 IC50 = 2140 nM T07279 CT2L4I 71512722 Ki = 900 nM T07279 CZR1K3 71533687 IC50 = 36 nM T07279 C1SM3T 71539661 Ki = 0.04 nM T07279 CX4JZ9 71547606 IC50 > 5000 nM T07279 C2T8KH 71547773 IC50 = 262 nM T07279 CCN01X 71547862 IC50 = 73 nM T07279 CIRD52 71547864 IC50 = 250 nM T07279 CM26ER 71547948 IC50 = 95 nM T07279 CC34DW 71547950 IC50 = 150 nM T07279 CA3O6K 71552696 IC50 = 14110 nM T07279 C1NPL0 71552941 IC50 > 30000 nM T07279 CA4PS8 71552942 IC50 > 30000 nM T07279 C6AN7B 71624486 Ki = 31 nM T07279 CJ4S3H 71624487 Ki = 2.8 nM T07279 CL5SN0 71624488 Ki = 7.8 nM T07279 C06VMT 71624600 Ki = 0.076 nM T07279 CRP0B1 71624601 Ki = 1.3 nM T07279 CEA49N 71624602 Ki = 0.52 nM T07279 CG16LA 71624603 Ki = 0.17 nM T07279 C7AOZ0 71624604 Ki = 0.65 nM T07279 C7L6CY 71624710 Ki = 18 nM T07279 CQ8AR2 71624711 Ki = 5.9 nM T07279 CEFO84 71624712 Ki = 4.9 nM T07279 CWK48Z 71624713 Ki = 0.094 nM T07279 CY52PM 71624822 Ki = 0.037 nM T07279 CGY4Z5 71730239 IC50 = 0.5 nM T07279 CS2RT7 71730241 IC50 = 1 nM T07279 CEZ0Y3 71730242 IC50 = 1.8 nM T07279 CR80EU 71730367 IC50 = 0.9 nM T07279 C09BGX 71731146 IC50 = 0.6 nM T07279 C5ES1L 71731394 IC50 = 2 nM T07279 CC2UI1 71731515 IC50 = 0.3 nM T07279 C87XSZ 71731781 IC50 = 0.1 nM T07279 C8VPO2 71731919 IC50 = 8.1 nM T07279 CCGY76 72545755 IC50 = 190 nM T07279 CET5H3 72545756 IC50 = 157 nM T07279 CK1IP9 72545757 IC50 = 1462 nM T07279 CZ94IO 72545758 IC50 = 87 nM T07279 CGH65P 72545759 IC50 = 781 nM T07279 CZ1P8N 72545761 IC50 = 2302 nM T07279 C4TWP5 72545996 IC50 = 4308 nM T07279 CV0T5B 72545997 IC50 = 114 nM T07279 CES3X4 72545998 IC50 = 212 nM T07279 CED7S2 72545999 IC50 = 19 nM T07279 CQG0D7 72546000 IC50 = 24 nM T07279 CJH0D1 72546229 IC50 = 137 nM T07279 CL0F6B 72546232 IC50 = 89 nM T07279 C9E4XZ 72546233 IC50 = 7.3 nM T07279 CFZS35 72546235 IC50 = 886 nM T07279 CW3C1O 72696648 IC50 = 3620 nM T07279 CFWX79 72696775 IC50 > 5000 nM T07279 CA21RI 72696776 IC50 = 3120 nM T07279 C4O7BN 72696777 IC50 = 4470 nM T07279 CIWC01 72696778 IC50 = 1315 nM T07279 CE1VB4 72696779 IC50 = 675 nM T07279 C83EPX 72696908 IC50 = 2222 nM T07279 CY0DG1 72696909 IC50 = 2406 nM T07279 CL4RD1 72696910 IC50 > 5000 nM T07279 C1A6VK 72696912 IC50 = 97 nM T07279 CY5AR8 72696914 IC50 = 502 nM T07279 C49GBP 72696916 IC50 = 184 nM T07279 C4GLH1 72697053 IC50 = 252 nM T07279 CJEC10 72697054 IC50 = 516 nM T07279 CC1H2R 72697055 IC50 = 684 nM T07279 CUCG27 72697056 IC50 = 275 nM T07279 C1HB3Q 72697057 IC50 = 956 nM T07279 C1LOH7 72697202 IC50 = 132 nM T07279 C62JGC 72715291 Ki = 0.44 nM T07279 C6H7QA 72725546 Ki = 6300 nM T07279 CJ15KC 72725547 Ki > 12500 nM T07279 CQ5K4U 72725607 Ki = 122 nM T07279 CVF34X 73056835 IC50 = 0.5 nM T07279 CVY2Z3 73056836 IC50 = 0.4 nM T07279 C25CJV 73057145 IC50 = 0.2 nM T07279 CHZ9U3 73352003 Ki = 21 nM T07279 C8MZG3 73354147 IC50 = 185 nM T07279 CXZ9J0 73356528 Ki = 2 nM T07279 CVF5P0 73603034 Ki = 0.1 nM T07279 CU5K6Q 74983184 Ki = 0.2 nM T07279 CYRP53 76310130 Ki > 12500 nM T07279 C49LJQ 76317357 Ki > 12500 nM T07279 CXZ30Q 76321071 Ki > 12500 nM T07279 CX4KN2 76331961 Ki = 7000 nM T07279 CXG04C 76331962 Ki > 12500 nM T07279 CJER97 76331963 Ki > 12500 nM T07279 CJ2T9E 76332983 IC50 > 10000 nM T07279 C0AYU9 76335538 Ki > 12500 nM T07279 C28YJW 76335539 Ki > 12500 nM T07279 C24USN 77050662 Ki = 0.11 nM T07279 CROJ27 78103829 Ki = 0.05 nM T07279 CGDC06 86294715 IC50 = 110 nM T07279 C3AF2E 86676680 Ki = 6000 nM T07279 C30ZNQ 86681992 IC50 = 420 nM T07279 CB7OC1 86681995 IC50 = 140 nM T07279 C5C1PH 86681998 IC50 = 510 nM T07279 CK8V3O 86725098 IC50 = 2710 nM T07279 C5R4CY 87057584 IC50 = 31 nM T07279 C4GF2R 89157636 IC50 = 99 nM T07279 CI57QV 89782019 IC50 = 0.38 nM T07279 CAG7B6 89782150 IC50 = 0.09 nM T07279 CH8JN1 89783250 IC50 = 0.1 nM T07279 C1CL8I 89783341 IC50 = 0.1 nM T07279 CUNJ79 89783434 IC50 = 0.3 nM T07279 CRQM10 89783564 IC50 = 2 nM T07279 CPX3K8 89783643 IC50 = 0.12 nM T07279 C2K3DA 89783801 IC50 = 0.38 nM T07279 CPQ9L3 89783993 IC50 = 0.3 nM T07279 C16ZQO 89784003 IC50 = 1 nM T07279 CDCO54 89784354 IC50 = 2 nM T07279 C8X1VA 89784686 IC50 = 0.13 nM T07279 CX2H4B 89784954 IC50 = 6.1 nM T07279 C0JIS8 89793954 IC50 = 117 nM T07279 C3N2TQ 89914568 Ki = 0.23 nM T07279 CXF3T0 90058666 IC50 = 0.08 nM T07279 C1UJ8Q 90058675 IC50 = 0.2 nM T07279 CWRJ32 90058676 IC50 = 0.5 nM T07279 CYZ98S 90058679 IC50 = 0.3 nM T07279 CFH4L6 90058683 IC50 = 0.05 nM T07279 CV9KG7 90058690 IC50 = 0.05 nM T07279 CP13IU 90058693 IC50 = 1 nM T07279 C56AJL 90058786 IC50 = 1 nM T07279 C35WJR 90058791 IC50 = 0.07 nM T07279 CCA78J 90058814 IC50 = 0.2 nM T07279 CN6H2I 90058905 IC50 = 0.4 nM T07279 C7DVW3 90058906 IC50 = 0.3 nM T07279 CYW61R 90256619 IC50 = 10 nM T07279 CK79BW 90256983 IC50 = 42 nM T07279 CX8NV6 90257109 IC50 = 1290 nM T07279 CX4J8N 90286701 IC50 > 10000 nM T07279 C75FLG 90326903 IC50 = 0.31 nM T07279 CN0V6L 90326906 IC50 = 1 nM T07279 CEV5P2 90645195 IC50 = 3130 nM T07279 C3E6PB 90656756 IC50 = 740 nM T07279 C95SGV 90656757 IC50 = 380 nM T07279 C0MWE6 90656758 IC50 = 590 nM T07279 CR3J7I 90656759 IC50 = 540 nM T07279 CHK6P8 90656760 IC50 = 660 nM T07279 CI68DP 90656761 IC50 = 310 nM T07279 COC3M0 90656762 IC50 = 630 nM T07279 C7JM5Z 90656763 IC50 = 920 nM T07279 C3MQ1Z 90656764 IC50 = 180 nM T07279 C5N1VZ 102581295 IC50 > 10000 nM T07279 C0A2RY 118720249 IC50 = 250 nM T07279 C95FJY 118720250 IC50 = 3600 nM T07279 C06XZY 118720251 IC50 = 4200 nM T07279 CVK71Z 118720252 IC50 = 180 nM T07279 C3CB8J 118720253 IC50 = 190 nM T07279 CV3ZY2 118720254 IC50 > 10000 nM T07279 CNI0U1 118720255 IC50 = 1900 nM T07279 CIX9N3 118720917 IC50 = 3730 nM T07279 CH09OX 118720918 IC50 = 1970 nM T07279 CVM73U 118721227 IC50 = 1640 nM T07279 CXY1K0 118721228 IC50 = 564 nM T07279 CEHY81 118725601 IC50 = 10 nM T07279 C6J7VS 118725602 IC50 = 16 nM T07279 CRY0X4 118725603 IC50 = 204 nM T07279 CY4P9O 118725604 IC50 = 1.3 nM T07279 CAT0C1 118725605 IC50 = 4.3 nM T07279 CL6CM1 118725606 IC50 = 6 nM T07279 C6JNB7 118725607 IC50 = 5 nM T07279 CE3B5A 118725608 IC50 = 6 nM T07279 C36FLX 118725609 IC50 = 4 nM T07279 CG6I4T 118725610 IC50 = 8 nM T07279 CN82QT 118725611 IC50 = 0.4 nM T07279 CUN73P 118725613 IC50 = 0.6 nM T07279 CL5K0U 118725614 IC50 = 1.5 nM T07279 CXEP50 118725615 IC50 = 0.6 nM T07279 CTUD48 118725865 IC50 > 22000 nM T07279 C5EH2L 122196349 Ki = 82 nM T07279 CKR45A 122196350 Ki = 0.17 nM T07279 CIF59P 122196351 Ki = 1.7 nM T07279 C2ES7U 122196352 Ki = 3900 nM T07279 C4I2VM 122196353 Ki = 2700 nM T07279 CZD9W8 123518123 IC50 = 9940 nM T07279 C0T6VF 123561371 IC50 = 5530 nM T07279 C04QEN 123616291 Ki = 0.3 nM T07279 C7G6IA 123944769 IC50 = 3590 nM T07279 CDL2V4 124005596 IC50 = 3010 nM T07279 C4ZS6N 127032072 Ki < 3 nM T07279 C1G4ES 127041542 Ki < 3 nM T07279 C8K0WU 127042183 Ki < 3 nM T07279 CC1VO7 127047444 IC50 = 730 nM T07279 CU95YJ 127050291 IC50 = 590 nM T07279 CFKY32 129012056 IC50 > 30000 nM T07279 C0FM1R 130196825 IC50 = 177 nM T07279 C4Q5LF 132471857 IC50 = 1400 nM T07279 C39UCD 133080605 IC50 = 6 nM T07279 C1W4DO 134135721 IC50 = 1.3 nM T07279 C9Z3XH 134138985 IC50 = 314 nM T07279 CX3A0W 134146922 IC50 = 0.09 nM T07279 CGBZ13 134843302 IC50 = 22000 nM T07279 CU60YC 135431661 IC50 = 1720 nM T07279 CSNE45 135461314 IC50 = 2963 nM T07279 C2UO7P 135566502 Ki = 2 nM T07279 CFN90Y 135566503 Ki = 29 nM T07279 CY4D8I 135566504 Ki = 164.2 nM T07279 C5DOH6 135566645 IC50 = 781 nM T07279 CN6E1U 135566647 IC50 = 197 nM T07279 CH2YR7 135566648 IC50 = 121 nM T07279 CN2B3D 135747628 IC50 = 0.05 nM T07279 CA6EQ3 135856841 Ki = 3 nM T07279 CO32WX 135856854 Ki = 63 nM T07279 C4X7QD 135856859 Ki = 149 nM T07279 C78FMI 135856860 Ki = 1250 nM T07279 CCJR27 135856881 Ki > 1424 nM T07279 C1CN9W 135856896 Ki = 206 nM T07279 CPL2Q0 135856897 Ki = 36 nM T07279 CLYW16 135856902 Ki = 16 nM T07279 CR8S9H 135856912 Ki = 153 nM T07279 CO47YW 135856913 Ki = 399 nM T07279 C39TEH 135856921 Ki = 211 nM T07279 CK9M5H 135867902 IC50 = 503 nM T07279 C20HYR 135867903 IC50 = 850 nM T07279 CZ70TA 135867906 IC50 = 653 nM T07279 C0MSR4 135867912 IC50 = 1068 nM T07279 CGM17H 135867918 IC50 = 1451 nM T07279 CUQ51Z 135867923 IC50 = 858 nM T07279 C0J7RQ 135867925 IC50 = 620 nM T07279 CORN45 135867927 IC50 = 840 nM T07279 CEX54P 135867940 IC50 = 72 nM T07279 C4XA7O 135867941 IC50 = 49 nM T07279 C8MR6U 135867952 IC50 = 5000 nM T07279 C0M9LS 135867953 IC50 = 2330 nM T07279 CP1VS6 135867954 IC50 = 5000 nM T07279 CIV27R 135867956 IC50 = 3330 nM T07279 CN8PW9 135867959 IC50 = 5000 nM T07279 CWSI79 135867966 IC50 = 3755 nM T07279 CTPK14 135867967 IC50 = 2377 nM T07279 CXU39R 135867972 IC50 = 3934 nM T07279 C2CZ9L 135867976 IC50 = 1741 nM T07279 CDYQ36 135867981 IC50 = 730 nM T07279 CP56XU 135867984 IC50 = 480 nM T07279 C28JUY 135867996 IC50 = 5000 nM T07279 C1GBJ8 135867997 IC50 = 598 nM T07279 CC92BK 135867998 IC50 = 293 nM T07279 C6RU2Z 135868002 IC50 = 3429 nM T07279 CK2EH9 135921041 Ki = 60 nM T07279 CW0XS9 135927905 Ki = 410 nM T07279 CB0X1D 135927906 Ki = 238 nM T07279 C97XNC 135927907 Ki > 1424 nM T07279 CCEL26 135927908 Ki = 147 nM T07279 C3G8VW 135927909 Ki > 1424 nM T07279 C3YD9J 135927910 Ki > 1424 nM T07279 CS9VK5 135927911 Ki = 122 nM T07279 CZ53AS 135927912 Ki = 83 nM T07279 CEI85B 135927919 Ki = 138 nM T07279 CB5N8A 135927920 Ki = 109 nM T07279 CCV12A 135927921 Ki = 13 nM T07279 C42TUA 135927922 Ki = 32 nM T07279 C1AJ7H 135927923 Ki = 21 nM T07279 CGUR31 135927924 Ki = 2 nM T07279 CG34TQ 135927925 Ki = 13 nM T07279 CIW7F3 135927928 Ki = 2 nM T07279 CX1B7W 135927929 Ki = 7 nM T07279 CWX70K 135927931 Ki = 84 nM T07279 C7HER4 135927932 Ki > 1424 nM T07279 CXOE95 135927933 Ki > 1424 nM T07279 CZOK96 135927935 Ki = 45 nM T07279 C34ZBN 135927936 Ki = 711 nM T07279 C47RLS 135927937 Ki > 1424 nM T07279 CV3H7I 135927938 Ki = 40 nM T07279 C19LMJ 135927939 Ki = 21 nM T07279 CZ25EG 135927940 Ki = 34 nM T07279 C4M7IK 135927941 Ki = 30 nM T07279 CX9SA7 135927946 Ki = 8 nM T07279 C90WDM 135927947 Ki = 13 nM T07279 C7E1TR 135927948 Ki = 44 nM T07279 CEXC86 135927949 Ki = 4 nM T07279 COM4E6 135927950 Ki = 12 nM T07279 C3QTI7 135927951 Ki = 29 nM T07279 CKN37Q 135927952 Ki = 5 nM T07279 C7RLI0 135927958 Ki = 99 nM T07279 CK8Z5W 135927959 Ki = 22 nM T07279 CCX4E5 135927960 Ki > 1420 nM T07279 C0ZP1O 135927961 Ki = 3 nM T07279 CP6W0X 135927962 Ki = 6 nM T07279 CPX81K 135927963 Ki = 3 nM T07279 C6F1QB 135927964 Ki = 66 nM T07279 CH1I0A 135927969 Ki = 2 nM T07279 C36KIX 135927970 Ki = 6 nM T07279 C28JYO 135927971 Ki = 152 nM T07279 C35IDA 135927972 Ki = 939 nM T07279 CN0J8C 135927973 Ki = 10 nM T07279 CG3UZ1 135927974 Ki = 2 nM T07279 C5E2KU 135927977 Ki = 120 nM T07279 C2OJK4 135927978 Ki = 29 nM T07279 C14JUY 135927979 Ki = 0.9 nM T07279 C1H2EG 135927980 Ki = 41 nM T07279 C7ZD2B 135928468 Ki = 23 nM T07279 C14OBQ 135928469 Ki = 3 nM T07279 C7C3MX 135928470 Ki = 5 nM T07279 CYTA89 135930672 IC50 = 194 nM T07279 CHA4N2 136013680 IC50 > 10 nM T07279 C3YL4I 136042193 IC50 = 1 nM T07279 CS4R2M 136098630 IC50 = 39 nM T07279 CWM2S3 136098631 IC50 = 283 nM T07279 CCB70U 136123533 Ki = 1140 nM T07279 CP3CA4 136189660 IC50 = 68 nM T07279 CC52HL 136189674 IC50 = 68 nM T07279 C4G9BI 136189695 IC50 = 68 nM T07279 CC87DY 136189770 IC50 = 5000 nM T07279 CTL8M5 136189797 IC50 = 87 nM T07279 CX45QN 136189847 IC50 = 140 nM T07279 CTVX09 136189895 IC50 = 134 nM T07279 CFZT23 136189934 IC50 = 29 nM T07279 CV9N1O 136190017 IC50 = 142 nM T07279 CQ85IN 136190059 IC50 = 534 nM T07279 CX8TS5 136190062 IC50 = 110 nM T07279 CLW25G 136190081 IC50 = 5000 nM T07279 C1YUD0 136219394 IC50 > 10 nM T07279 CAY7U9 136236280 IC50 > 1000 nM T07279 C73IGY 136244208 IC50 = 29 nM T07279 CXS5Z6 136254223 IC50 = 5000 nM T07279 C2DNM5 136254224 IC50 > 5000 nM T07279 CQM1U4 136254225 IC50 = 162 nM T07279 COU4C5 136254226 IC50 = 5000 nM T07279 CQU6J7 136254227 IC50 = 5000 nM T07279 CIU8W3 136254389 IC50 > 10 nM T07279 C3MK9W 136807986 IC50 > 10000 nM T07279 C4VAQ0 136966273 IC50 = 0.7 nM T07279 CVG90R 137631416 IC50 = 15 nM T07279 CYQJ28 137632388 IC50 = 116 nM T07279 CV1A5N 137633544 IC50 = 872 nM T07279 CI1E8V 137634241 IC50 > 10000 nM T07279 C6D8IM 137634495 IC50 = 1270 nM T07279 CK7QM8 137634713 Ki = 630 nM T07279 C9AIT8 137634969 IC50 = 300 nM T07279 CA1D9B 137636162 IC50 = 640 nM T07279 CF65JZ 137636187 IC50 = 140 nM T07279 CD5IZ6 137636389 Ki = 16 nM T07279 CSQ0T2 137636417 IC50 = 16 nM T07279 CQ5S9H 137636735 IC50 = 148 nM T07279 CU9YQ3 137637635 IC50 > 10000 nM T07279 C5HD0W 137638179 IC50 = 6 nM T07279 C1MO4H 137638461 IC50 = 34 nM T07279 CUF1D9 137638752 Ki = 9.6 nM T07279 C21XCP 137638981 IC50 = 24 nM T07279 CJ69GR 137638996 IC50 = 99 nM T07279 CV5M4H 137640638 IC50 = 290 nM T07279 C25JLY 137640893 IC50 = 135 nM T07279 CI0NF6 137641367 IC50 > 30000 nM T07279 C30DWC 137642509 Ki = 170 nM T07279 CPO2G4 137642902 IC50 = 89 nM T07279 CHD90A 137643257 Ki = 13 nM T07279 C2MO5L 137643556 IC50 = 383 nM T07279 CHOI53 137643582 IC50 = 22 nM T07279 CNL3U7 137643747 IC50 = 298 nM T07279 CL6K4E 137643873 IC50 = 3300 nM T07279 CJS20N 137644367 IC50 = 9 nM T07279 C0DAH4 137644542 IC50 = 660 nM T07279 CB2Z5V 137646513 IC50 = 1950 nM T07279 C1H3ZK 137647783 IC50 = 6 nM T07279 C3JDR6 137648580 Ki = 18 nM T07279 C7UTE8 137648598 IC50 = 13 nM T07279 CCZE58 137650076 IC50 = 25 nM T07279 CAK39E 137650557 IC50 = 4220 nM T07279 CDF3Q7 137650805 IC50 > 30000 nM T07279 C8J3RF 137651484 IC50 = 28 nM T07279 C2EA4F 137652505 IC50 = 15 nM T07279 C4CWB2 137654577 IC50 = 57 nM T07279 CIZ8M6 137654684 IC50 = 109 nM T07279 CSQG93 137654724 IC50 = 23 nM T07279 CZE82A 137655925 IC50 = 10 nM T07279 CFXC14 137656007 Ki = 0.48 nM T07279 C1BEV7 137656991 IC50 = 99 nM T07279 CF25MB 137659327 IC50 = 6 nM T07279 C72ZDI 137659673 Ki = 7.9 nM T07279 C70GPH 137659881 IC50 = 179 nM T07279 C4OUD0 137660252 Ki = 7400 nM T07279 CW57TM 137661945 IC50 = 7410 nM T07279 CQ82UE 137662204 IC50 > 30000 nM T07279 CS32YP 145960484 IC50 = 770 nM T07279 CHZ20V 145960670 IC50 > 10000 nM T07279 C81DKZ 145960765 IC50 = 1380 nM T07279 C8M2RY 145960938 IC50 = 650 nM T07279 CNSO87 145961054 IC50 = 537 nM T07279 CD2O0Q 145961184 IC50 = 460 nM T07279 CY25XU 145961279 IC50 = 700 nM T07279 C8IAB5 145961349 IC50 = 2160 nM T07279 CDTI85 145961440 IC50 = 820 nM T07279 CXU40G 145961470 IC50 = 259 nM T07279 CW15YM 145961475 IC50 > 10000 nM T07279 CUI86V 145961560 IC50 = 2120 nM T07279 CE26LP 145961625 IC50 = 5330 nM T07279 CV15YW 145961659 IC50 = 230 nM T07279 C0KY1T 145961724 IC50 > 10000 nM T07279 C2YQF0 145961914 IC50 = 2260 nM T07279 CH2V4T 145961915 IC50 = 370 nM T07279 CQLA92 145961972 IC50 = 841 nM T07279 COW23H 145962040 IC50 = 870 nM T07279 C7OF6V 145962094 IC50 = 220 nM T07279 CB3O4I 145962109 IC50 > 10000 nM T07279 CP3EH0 145962188 IC50 = 645 nM T07279 C9S8AO 145962192 IC50 = 560 nM T07279 CZIT45 145962335 IC50 = 2540 nM T07279 CTN2B1 145962545 IC50 = 4320 nM T07279 C5NCH1 145962614 IC50 > 10000 nM T07279 C2TRN8 145962743 IC50 = 7950 nM T07279 CLS90K 145962852 IC50 = 2780 nM T07279 CJD24A 145962897 IC50 = 1620 nM T07279 C9C3YP 145962963 IC50 = 5800 nM T07279 C69ZIQ 145963064 IC50 > 10000 nM T07279 C01JIP 145963077 IC50 > 10000 nM T07279 CJQ78W 145963108 IC50 = 4350 nM T07279 CY8RS4 145963277 IC50 = 4440 nM T07279 CUI0L7 145963307 IC50 = 1426 nM T07279 CO4Y1M 145963467 IC50 = 267 nM T07279 C8QDJ0 145963511 IC50 > 10000 nM T07279 C1J5BC 145963517 IC50 = 830 nM T07279 C3TLW0 145963725 IC50 = 1800 nM T07279 CV28AL 145967603 IC50 > 30000 nM T07279 C5B0QL 145967935 IC50 = 26000 nM T07279 CMG01Q 145968043 IC50 > 30000 nM T07279 C9LBY8 145968158 IC50 > 30000 nM T07279 CPET15 145968269 IC50 > 30000 nM T07279 C24AQX 145968504 IC50 > 30000 nM T07279 CTY0I5 145968604 IC50 > 30000 nM T07279 CL07SI 145968637 IC50 = 22000 nM T07279 C7B3UD 145968656 IC50 = 6900 nM T07279 CZN38I 145969224 IC50 > 30000 nM T07279 CL8V5N 145969695 IC50 > 30000 nM T07279 CAU16Y 145969796 IC50 > 30000 nM T07279 CISA20 145969798 IC50 > 30000 nM T07279 CM6D9P 145969896 IC50 > 30000 nM T07279 CT3N9K 145970124 IC50 > 30000 nM T07279 CQR9Z4 145970125 IC50 = 10000 nM T07279 CP0M6D 145970925 IC50 > 30000 nM T07279 CQ4WO3 145971039 IC50 = 2800 nM T07279 CD97BO 145971046 IC50 > 30000 nM T07279 C09DLU 145971051 IC50 > 30000 nM T07279 C4P8SD 145989719 IC50 = 140 nM T07279 CYGN68 155510554 IC50 = 4250 nM T07279 C25TBW 155511840 IC50 = 0.83 nM T07279 CC1V3X 155511863 IC50 = 0.12 nM T07279 C2MD1Q 155513187 IC50 > 10000 nM T07279 CDF0I2 155514882 IC50 = 4870 nM T07279 C7BMF4 155515543 IC50 = 0.08 nM T07279 C4RFU7 155516598 IC50 = 1.6 nM T07279 CU35GB 155517528 IC50 = 29.4 nM T07279 CS3E7L 155518082 IC50 = 2.2 nM T07279 CY49NZ 155518625 IC50 = 6.7 nM T07279 C24NBM 155518799 IC50 = 0.18 nM T07279 C4T6CH 155518837 IC50 = 1930 nM T07279 CO58XZ 155519799 IC50 = 2.7 nM T07279 CKD52G 155520766 IC50 = 8040 nM T07279 CJ5L2U 155520986 Ki = 9 nM T07279 CV42MB 155521123 IC50 = 0.15 nM T07279 CM8HF6 155521436 Ki = 0.3 nM T07279 CGQH30 155523583 Ki = 0.2 nM T07279 CUM08K 155524352 IC50 = 0.16 nM T07279 CQ0I3P 155524597 IC50 > 10000 nM T07279 C3BTZ8 155525211 Ki = 6 nM T07279 CY7EM6 155525492 IC50 = 15.7 nM T07279 CX59UT 155526046 IC50 = 4 nM T07279 CE5ZU0 155526194 IC50 = 1270 nM T07279 CQ4XA9 155527433 IC50 = 122 nM T07279 C5OBZ9 155527556 Ki = 0.04 nM T07279 C76QNG 155528354 IC50 = 2470 nM T07279 CR5ON6 155528414 IC50 = 0.13 nM T07279 C2R8JO 155528784 IC50 > 1000 nM T07279 CN0M8O 155529692 IC50 = 3.2 nM T07279 CEF14U 155529807 IC50 = 0.7 nM T07279 CS9W1N 155531462 IC50 = 11 nM T07279 C2N6XM 155531935 IC50 = 4690 nM T07279 CY59IV 155531989 IC50 = 6 nM T07279 C8IP7E 155532982 IC50 = 2870 nM T07279 C3K2ZL 155533051 IC50 = 0.24 nM T07279 CIH5W7 155534088 IC50 = 0.18 nM T07279 CL7U8D 155534608 IC50 = 5.7 nM T07279 CF65PU 155535300 IC50 = 0.11 nM T07279 CQ97VC 155535921 IC50 = 0.6 nM T07279 C68GMW 155538446 IC50 > 10000 nM T07279 CX90PO 155538459 IC50 = 0.41 nM T07279 C6QY8K 155538969 IC50 = 0.16 nM T07279 C9J3IU 155538981 IC50 = 6210 nM T07279 C68KHN 155539424 IC50 = 6.8 nM T07279 CXV14T 155539760 IC50 = 696 nM T07279 C4H0LS 155541271 IC50 = 4010 nM T07279 CWQ7F0 155541490 IC50 = 7.4 nM T07279 CY8PB1 155542894 IC50 = 1100 nM T07279 C2IG7U 155543022 IC50 = 2.1 nM T07279 CE03IU 155543981 IC50 > 10000 nM T07279 CRG0K4 155544306 IC50 = 2.5 nM T07279 CPB87M 155545130 IC50 = 10.2 nM T07279 CNL4B8 155546196 IC50 = 7.4 nM T07279 CC83QJ 155547453 IC50 = 21 nM T07279 CEDN41 155550408 IC50 = 5.1 nM T07279 CB73CQ 155551312 IC50 = 10.4 nM T07279 CG26ND 155552144 IC50 = 5.2 nM T07279 CORH39 155553574 IC50 = 3330 nM T07279 CH18PL 155553803 IC50 = 5530 nM T07279 CY6Q8S 155554337 IC50 > 10000 nM T07279 CXO5L1 155556907 IC50 = 27 nM T07279 C6CJ3H 155557017 IC50 = 1.1 nM T07279 C62DJU 155558058 IC50 = 4.9 nM T07279 CU1MA5 155558576 IC50 = 1650 nM T07279 CM0UH7 155559265 IC50 = 17.5 nM T07279 C95EJG 155559459 IC50 = 0.16 nM T07279 CO2I4P 155559898 IC50 = 11000 nM T07279 CG6T9Y 155559978 IC50 = 858 nM T07279 CRLP86 155560079 IC50 = 9 nM T07279 CJ9M3Y 155563039 IC50 = 0.6 nM T07279 C4EX3W 155563397 IC50 = 3.5 nM T07279 C46LPJ 155563540 IC50 = 3740 nM T07279 C43CBF 155566090 IC50 = 6.1 nM T07279 C9WB2L 155566373 IC50 = 9.9 nM T07279 C1B7YH 155566566 IC50 = 0.9 nM T07279 C04THL 155567360 IC50 = 6.1 nM T07279 C4ED0G 155568443 IC50 = 1 nM T07279 CTZ24C 155568643 IC50 = 0.23 nM T07279 CV8W5R 155569485 IC50 = 9.3 nM T07279 D00ERW 44444843 Ki > 1424 nM T07279 D00HVA 11624601 Ki > 1400 nM T07279 D06HVH 54613583 IC50 = 240 nM T07279 D06UKS 44222958 IC50 = 6 nM T07279 D07DJS 5280459 IC50 = 25000 nM T07279 D07OXC 11650194 IC50 > 25000 nM T07279 D09HVH 135566652 IC50 > 10 nM T07279 D09OWC 5373936 IC50 = 300 nM T07279 D0Q3NG 11715520 Ki > 1400 nM T07279 D0S7IE 11658882 Ki > 1400 nM T27466 CG3PR6 52912222 IC50 > 1 nM T27466 CIPN50 71760902 IC50 > 10000 nM T27466 C5TB9S 77843982 IC50 > 10000 nM T27466 COZ8S1 78319129 IC50 > 10000 nM T27466 CF9J8E 118918705 IC50 = 190 nM T27466 CA3Z8O 118918714 IC50 = 1000 nM T27466 C8GLJ3 118918720 IC50 = 2300 nM T27466 CAZR96 118918740 IC50 = 10000 nM T27466 C2ZY3U 118932975 IC50 = 2200 nM T27466 CHCU32 118932979 IC50 = 2200 nM T27466 C2JCY3 118932989 IC50 = 2200 nM T27466 CC14FI 118933132 IC50 = 260 nM T27466 CEPT12 118933133 IC50 = 280 nM T27466 CKY8H3 118933134 IC50 = 590 nM T27466 CGO91Y 118933136 IC50 = 9300 nM T27466 CBD7I6 121232405 IC50 = 15848.93 nM T27466 CWJD15 122705990 IC50 = 2450 nM T27466 CG9S7A 126961735 Ki = 100 nM T27466 CED70X 130472274 IC50 > 20000 nM T27466 CK0B6N 131985884 IC50 = 7600 nM T27466 CPWF20 137632687 IC50 = 4600 nM T27466 CD4NE1 137633137 IC50 = 4600 nM T27466 CQT3A9 137636309 IC50 > 100000 nM T27466 CV1EP8 137639742 IC50 > 100000 nM T27466 CC3VL8 137644086 IC50 = 16000 nM T27466 CC34KQ 137650533 IC50 = 12000 nM T27466 CQ6XB7 139030526 IC50 = 10000 nM T27466 D03BTJ 15990224 IC50 > 100000 nM T27466 D0C2PD 50796983 IC50 = 7000 nM T27466 D0O6XT 91827373 IC50 = 140 nM T27466 D0Q7IU 40642506 IC50 = 5110 nM T00254 C6BM3N 50916706 EC50 = 100 nM T00254 C2AY0O 50925116 EC50 = 1100 nM T00254 CGF2A0 57394020 IC50 = 670 nM T00254 CTD0E1 57394021 IC50 = 790 nM T00254 CRKJ42 60168095 EC50 = 650 nM T00254 C27CXW 60168096 EC50 > 3000 nM T00254 C3ME9Z 60168097 EC50 = 140 nM T00254 C73KDV 60168098 EC50 = 77 nM T00254 CU97LH 70681530 EC50 > 3000 nM T00254 CV56DC 70682168 EC50 = 3000 nM T00254 CS2T0P 70682169 EC50 = 800 nM T00254 C3J4BU 70682171 EC50 = 7400 nM T00254 C8HBM7 70682172 EC50 = 1600 nM T00254 C3C9QW 70682182 EC50 = 630 nM T00254 CYMX54 70683637 EC50 = 2500 nM T00254 CLOD09 70683638 EC50 = 1700 nM T00254 CJ8I3A 70683652 EC50 = 780 nM T00254 C35HZS 70684281 EC50 = 3000 nM T00254 C2IO8X 70684282 EC50 = 7800 nM T00254 C7UE6D 70684283 EC50 = 2600 nM T00254 CPJ42Z 70684284 EC50 = 2500 nM T00254 C32TLG 70684287 EC50 = 670 nM T00254 CFIJ16 70685790 EC50 = 1200 nM T00254 C36UDB 70685792 EC50 = 97 nM T00254 C3KRS9 70685793 EC50 = 2000 nM T00254 C3T7BQ 70685794 EC50 = 710 nM T00254 CC9X5Z 70686432 EC50 = 2000 nM T00254 C4GTQ5 70686433 EC50 = 3900 nM T00254 CBYT67 70687909 EC50 = 840 nM T00254 C89SZF 70687919 EC50 = 600 nM T00254 CE06PD 70687920 EC50 = 330 nM T00254 CQ0Z9L 70688529 EC50 = 2500 nM T00254 CH6DC4 70688530 EC50 = 2500 nM T00254 CC05RM 70688531 EC50 = 2500 nM T00254 CL1KT9 70689938 EC50 = 2100 nM T00254 CY9EK4 70689939 EC50 > 3000 nM T00254 C30DRH 70692109 EC50 = 650 nM T00254 CQ56AT 70692734 EC50 = 2600 nM T00254 CFC42A 70692735 EC50 = 4000 nM T00254 C7CJ8W 70692745 EC50 = 400 nM T00254 C1HY6B 70692746 EC50 = 570 nM T00254 CG6C1S 70694153 EC50 = 120 nM T00254 CX5U0C 70694154 EC50 = 620 nM T00254 C7A6UB 70694774 EC50 = 2900 nM T00254 CS8RX9 70694775 EC50 = 8800 nM T00254 C6CBO5 70694776 EC50 = 5500 nM T00254 C10WHV 70694777 EC50 = 620 nM T00254 CIR89G 70694778 EC50 = 670 nM T00254 CD9J7R 70696280 EC50 = 800 nM T00254 CYF8G0 70696281 EC50 = 120 nM T00254 CP86JE 70696821 EC50 = 1800 nM T00254 CN9YI0 70696824 EC50 = 1600 nM T00254 C6XG5N 70696834 EC50 = 450 nM T00254 C70QOT 71682479 EC50 = 50 nM T00254 CAR09D 71682481 EC50 = 63 nM T00254 C1TB8G 71682483 EC50 = 160 nM T00254 C4SV3Z 71682624 EC50 = 160 nM T00254 C6MQ7J 71682626 EC50 = 160 nM T00254 CL04WU 71682627 EC50 = 160 nM T00254 CF0Y4S 71682629 EC50 = 200 nM T00254 C5O9HB 71682631 EC50 = 200 nM T00254 C6F8IQ 71682633 EC50 = 200 nM T00254 CBF79Z 71682784 EC50 = 400 nM T00254 CSJQ97 71682786 EC50 = 400 nM T00254 C0B1QU 71682787 EC50 = 200 nM T00254 CACO06 71682788 EC50 = 250 nM T00254 CQ39RJ 71682789 EC50 = 400 nM T00254 C5M2FV 71682790 EC50 = 630 nM T00254 CAV4K9 71682791 EC50 > 50000 nM T00254 CE8TN9 71682936 EC50 > 50000 nM T00254 C7LWD9 71682937 EC50 = 200 nM T00254 C7ZLE2 71682938 EC50 = 200 nM T00254 C0IQ5Y 71682939 EC50 = 630 nM T00254 CV96CP 71682940 EC50 = 630 nM T00254 C8C3DJ 71682941 EC50 > 50000 nM T00254 D07IZG 50905018 EC50 = 400 nM T56418 D01PZD 5329098 IC50 = 1200 nM T56418 D03ZBT 11626560 EC50 = 0.47 nM T56418 D04LVK 57379345 IC50 = 0.2 nM T56418 D08PIE 68165256 IC50 = 0.37 nM T56418 D0AF6O 71731823 Ki < 0.07 nM T56418 D0K8KX 5280343 IC50 = 3320 nM T56418 D0O8GK 71496458 IC50 = 177 nM T56418 D0R0MW 5329102 IC50 = 2300 nM T56418 D0U3SY 49806720 IC50 = 2.07 nM T56418 D01HKZ 57345941 IC50 = 1.2 nM T56418 D03HUX 49792852 IC50 > 10000 nM T56418 D03LWG 53235510 IC50 = 3078 nM T56418 D05NFR 135565923 IC50 = 1.01 nM T56418 D07EHV 44814409 IC50 > 10000 nM T56418 D07HPJ 11476171 IC50 > 5500 nM T56418 D08HOM 46207586 IC50 = 363 nM T56418 D0D1GF 42642645 IC50 > 3000 nM T56418 D0E3TC 44259 IC50 = 0.74 nM T56418 D0FD6D 11751922 IC50 = 132 nM T56418 D0KX7I 56960363 IC50 < 0.4 nM T56418 D0N6NM 71721648 IC50 = 22 nM T56418 D0O0LQ 11364421 IC50 = 180 nM T56418 D0O0LS 25141092 Ki = 6.2 nM T56418 D0O9PQ 57390074 IC50 = 0.07 nM T56418 D0P1CV 46191454 IC50 > 10000 nM T56418 D03BNU 59604787 IC50 > 3500 nM T56418 D0T3ME 156422 IC50 > 30000 nM T56418 CVS0R8 709497 IC50 = 2850 nM T56418 C5XK3N 719280 IC50 = 6460 nM T56418 CUTS74 719592 IC50 = 3750 nM T56418 COH21C 951145 IC50 = 4240 nM T56418 C1RQ4E 1886699 IC50 = 4000 nM T56418 C6NK9W 1898760 IC50 = 2100 nM T56418 CJ7L5Z 5124249 IC50 = 112000 nM T56418 C8IAR2 5281657 IC50 = 41300 nM T56418 CI68PW 5283685 IC50 = 4730 nM T56418 CXK0S6 5283727 IC50 = 7550 nM T56418 C0LS8P 5714573 IC50 = 1380 nM T56418 C4YJ3C 5714584 IC50 = 1730 nM T56418 CB7IH1 7200289 IC50 = 8660 nM T56418 C4G9WR 9547398 IC50 > 100000 nM T56418 C76CUP 9547698 IC50 = 4160 nM T56418 CN0AJ9 9934347 IC50 = 5 nM T56418 CR8DA1 10024683 IC50 > 100000 nM T56418 CLA93G 10047202 IC50 = 4360 nM T56418 C3LCH5 10047545 IC50 > 100000 nM T56418 CUJR40 10062694 EC50 > 2000 nM T56418 C7SFI1 10296883 IC50 > 10000 nM T56418 C4CP7K 10423452 IC50 = 1100 nM T56418 C7HBP6 10429593 IC50 > 10000 nM T56418 C83QWV 10714343 IC50 = 2190 nM T56418 C92JSF 10979489 IC50 = 910 nM T56418 C8G5WP 11210533 IC50 = 250 nM T56418 CLZ3M8 11442557 IC50 = 91 nM T56418 CQ06DZ 11532796 IC50 = 26800 nM T56418 CWHK97 11553173 IC50 = 19500 nM T56418 CKO0G8 11568821 IC50 > 40000 nM T56418 CMN1Q3 11569457 IC50 = 7500 nM T56418 CDT68P 11576099 IC50 = 5500 nM T56418 C5DHZ2 11590126 IC50 = 3000 nM T56418 C43JZU 11604436 Ki = 600 nM T56418 CGU7N0 11604739 Ki = 500 nM T56418 CYA04X 11605000 IC50 = 14500 nM T56418 CJ97KW 11655878 IC50 = 13800 nM T56418 CAJS96 11662893 Ki = 1100 nM T56418 CKAH36 11669784 Ki = 200 nM T56418 CJ9KN7 11683817 IC50 > 10000 nM T56418 C6EOL3 11691146 IC50 = 3700 nM T56418 CTRZ62 11705264 IC50 = 20300 nM T56418 CA2KE3 11719817 IC50 = 3800 nM T56418 CQN23V 15551239 IC50 = 4800 nM T56418 C5VPH9 16129448 IC50 = 266 nM T56418 COJR59 16910714 IC50 = 3470 nM T56418 CBD9U4 23647620 IC50 = 11000 nM T56418 CA3I4T 24753787 IC50 > 5000 nM T56418 CAJ4T2 24762205 IC50 > 10000 nM T56418 CN8R5S 24779728 IC50 = 15 nM T56418 C5YW7P 24825755 IC50 > 10000 nM T56418 C2PM9I 24852349 IC50 > 10000 nM T56418 CLT79V 24852790 IC50 = 256 nM T56418 C5LQC0 24853018 IC50 = 145 nM T56418 CP1DO3 24853225 IC50 = 15 nM T56418 CBAQ48 24853329 IC50 = 200 nM T56418 CY8L7E 24896769 IC50 > 10000 nM T56418 C4EG8R 24993189 IC50 > 10000 nM T56418 C4OA5D 25113170 IC50 = 0.5 nM T56418 CS9G4P 25157326 IC50 = 5 nM T56418 C3VR6L 25157614 IC50 = 20 nM T56418 C10CVP 25160012 IC50 = 25 nM T56418 CUAB05 25160153 IC50 = 14.6 nM T56418 CCM97P 25160155 IC50 = 43.5 nM T56418 C8IX5P 25174241 IC50 = 14 nM T56418 CTKC48 25174394 IC50 = 684 nM T56418 CE6PB7 25175712 IC50 = 73 nM T56418 CB1Z8N 25175860 IC50 = 67 nM T56418 CIHB16 25175861 IC50 = 30 nM T56418 CVO5B2 25175862 IC50 = 38 nM T56418 C04HDK 25176007 IC50 = 15 nM T56418 CT2K5R 25176014 IC50 = 3 nM T56418 C8A9EJ 25176163 IC50 = 560 nM T56418 C6G7RT 25176165 IC50 = 10 nM T56418 CPM9Q8 25176330 IC50 = 378 nM T56418 C81NBM 25176332 IC50 = 210 nM T56418 CI58TS 25176649 IC50 = 72 nM T56418 CSEN02 25176653 IC50 = 135 nM T56418 CM0T8S 25210970 IC50 = 0.4 nM T56418 CNQ9G5 25218180 IC50 < 1000 nM T56418 CO0RF6 25218593 IC50 = 1 nM T56418 CNJ3Y1 44181654 IC50 = 40 nM T56418 CF9UB1 44219665 IC50 > 40000 nM T56418 CXPN30 44219666 IC50 = 9300 nM T56418 CVEU45 44219667 IC50 = 6200 nM T56418 CR91QB 44480266 IC50 > 10000 nM T56418 C1NM5K 44481287 IC50 = 360 nM T56418 C4B7KF 44515722 IC50 = 0.18 nM T56418 C8H4FA 44515723 IC50 = 1.06 nM T56418 CUT5I7 44517769 IC50 = 0.6 nM T56418 C6OC4Z 44607530 IC50 = 990 nM T56418 CU3RF1 45139989 IC50 > 10000 nM T56418 CQGZ06 45139991 IC50 > 10000 nM T56418 C4K8BX 45267171 IC50 = 21300 nM T56418 C25VIM 45267176 IC50 = 18000 nM T56418 C7RF4H 45267177 IC50 = 8300 nM T56418 CV94UD 45268038 IC50 = 5800 nM T56418 C64DKR 45268916 IC50 = 7100 nM T56418 CRC85D 45270590 IC50 = 5000 nM T56418 C36DGY 45272290 IC50 > 40000 nM T56418 COT0W8 45272300 IC50 = 5100 nM T56418 CC79UA 45273165 IC50 = 11800 nM T56418 CNR8G6 45273175 IC50 > 40000 nM T56418 CF57GK 46215462 IC50 = 530 nM T56418 CKC04F 46220497 IC50 = 48 nM T56418 C85RJI 46233108 IC50 = 3800 nM T56418 C19SZF 46233185 IC50 > 50000 nM T56418 C7ON5A 46233287 IC50 > 10000 nM T56418 CL07DO 46838818 IC50 = 35000 nM T56418 CNW6I7 46838966 IC50 = 1700 nM T56418 C9DR6V 46838967 IC50 = 9700 nM T56418 CG24VC 46852202 IC50 = 11 nM T56418 CQL10H 46852353 IC50 > 2000 nM T56418 CO8N0C 46852969 IC50 = 91 nM T56418 C6JWM5 46871637 IC50 = 10 nM T56418 CLS29B 46872626 IC50 > 10000 nM T56418 C2R8LA 46906623 IC50 = 506 nM T56418 C0SXY7 46906669 IC50 = 11 nM T56418 CWG19F 46906670 IC50 = 465 nM T56418 CWL4N0 46906671 IC50 > 10000 nM T56418 C96QSL 46906672 IC50 > 10000 nM T56418 C54HJW 46906715 IC50 = 1538 nM T56418 C3FW0P 46906716 IC50 > 3000 nM T56418 CYU5K8 46906717 IC50 > 3000 nM T56418 CBSX87 46906718 IC50 = 1302 nM T56418 C7QDB9 46906792 IC50 = 121 nM T56418 C4OZD0 46906793 IC50 = 450 nM T56418 CJ8I6H 46906794 IC50 = 250 nM T56418 CF0U6S 46907265 IC50 = 27 nM T56418 CQ1SO3 46907305 IC50 = 278 nM T56418 C2B5XF 49765254 IC50 > 10000 nM T56418 C0SJ7Q 49804868 IC50 = 15.1 nM T56418 CF0NP4 49805004 IC50 = 1.8 nM T56418 COR4V2 49806718 IC50 = 2.4 nM T56418 C5ME3S 49806721 IC50 = 2.9 nM T56418 C67HGW 49806722 IC50 = 1.1 nM T56418 CJZ5A0 49840306 IC50 > 10000 nM T56418 CRA74I 49842779 IC50 = 3500 nM T56418 CF91RS 49843531 IC50 > 10000 nM T56418 CIA9Z7 50877838 IC50 = 59100 nM T56418 CBC62W 50899254 IC50 > 10000 nM T56418 C2Y6QS 50938552 IC50 > 10000 nM T56418 CF28WU 50939519 IC50 < 0.5 nM T56418 CP7B9V 50942696 IC50 = 4 nM T56418 C9NYP4 51036677 IC50 > 10000 nM T56418 C4WRY3 51037112 IC50 > 10000 nM T56418 CRI28Z 51037948 IC50 > 10000 nM T56418 CM24LF 52938983 IC50 = 2.71 nM T56418 CF20TR 53317353 IC50 = 49 nM T56418 C8QL7R 53317354 IC50 = 4 nM T56418 CMDP24 53317655 IC50 = 6 nM T56418 C5M3OC 53318635 IC50 = 7 nM T56418 C6Q8MV 53318636 IC50 = 10 nM T56418 CTG1Z2 53318637 IC50 = 6 nM T56418 CM0L9V 53319073 IC50 = 4 nM T56418 CA4I8S 53319963 IC50 = 120 nM T56418 CZ0BV7 53320342 IC50 > 10000 nM T56418 CK7A8Y 53321265 IC50 = 175 nM T56418 C9D8EB 53321266 IC50 = 65 nM T56418 CQD92F 53322588 IC50 = 5 nM T56418 C2W9OA 53324451 IC50 = 763 nM T56418 C3DO4U 53325211 IC50 = 58 nM T56418 CM7P3W 53357328 IC50 = 1.5 nM T56418 C4QO8D 53364164 IC50 = 3030 nM T56418 C8NA4L 53384644 IC50 > 30000 nM T56418 C24FQU 53465297 IC50 = 10 nM T56418 C67XFO 53482132 IC50 = 6 nM T56418 C5VG9P 53495177 IC50 = 16 nM T56418 CI12VS 54577678 IC50 = 38 nM T56418 COF6B0 54577892 IC50 = 20 nM T56418 C5TAL7 54577893 IC50 = 726 nM T56418 CPS75F 54577894 IC50 = 883 nM T56418 C17PKQ 54577895 IC50 = 260 nM T56418 C2ECL9 54577896 IC50 = 7 nM T56418 CZ9W6N 54577897 IC50 = 9 nM T56418 C08ABD 54578104 IC50 = 5 nM T56418 CIV58E 54578105 IC50 = 3.8 nM T56418 C0W4QA 54578108 IC50 = 9 nM T56418 C0KI7N 54578323 IC50 = 15 nM T56418 COEX71 54578324 IC50 = 7 nM T56418 CKAP47 54578772 IC50 = 27 nM T56418 CR9F8Q 54578773 IC50 = 10.6 nM T56418 C4Z1NO 54578774 IC50 = 2.7 nM T56418 CD6RH1 54578996 IC50 = 66.4 nM T56418 CV79SW 54578997 IC50 = 186 nM T56418 C9S4RT 54580866 IC50 = 40 nM T56418 CR5AF2 54580867 IC50 = 7.6 nM T56418 CT50VL 54580868 IC50 = 11.4 nM T56418 C0W7RC 54581811 IC50 = 367.6 nM T56418 CM70UI 54581812 IC50 = 89.1 nM T56418 CFML47 54582849 IC50 = 80 nM T56418 CLT2S9 54582850 IC50 = 26.2 nM T56418 CN0GR2 54583855 IC50 = 2470 nM T56418 CL7BT1 54583856 IC50 = 660 nM T56418 CU51TS 54584736 IC50 = 9290 nM T56418 CBJ4V1 54584737 IC50 = 61.8 nM T56418 C05KTP 54584738 IC50 = 50.8 nM T56418 C7RD1A 54584739 IC50 = 68.3 nM T56418 C37SZJ 54584802 Ki = 170 nM T56418 C4NGT9 54584814 IC50 = 770 nM T56418 CT87JD 54584815 IC50 = 3.7 nM T56418 CX7U6B 54585675 IC50 = 604.5 nM T56418 CLV6D8 54585676 IC50 = 415.3 nM T56418 CET3M2 54586749 IC50 = 2080 nM T56418 CEZ37O 54586750 IC50 = 850 nM T56418 C0A3VW 54586751 IC50 = 11.6 nM T56418 C70NRJ 54586752 IC50 = 33.4 nM T56418 CVS20L 54586753 IC50 = 37.4 nM T56418 C37RNP 54587692 IC50 = 149.3 nM T56418 CM20ZP 54587775 IC50 = 3470 nM T56418 C7NLB8 54587776 IC50 = 100 nM T56418 CKY7E4 54587777 IC50 = 18.5 nM T56418 C70KGE 54588490 Ki = 0.4 nM T56418 CT71UH 54596950 IC50 = 10 nM T56418 C2F6DB 54596952 IC50 = 19 nM T56418 CXO6Y4 54597025 IC50 = 28 nM T56418 C8AB1J 54759606 Ki = 95 nM T56418 C1XS2J 54760383 IC50 = 2300 nM T56418 C69FXM 54760600 IC50 = 14 nM T56418 C9ZFS1 54764923 IC50 = 9330 nM T56418 CRH20S 56596558 IC50 = 174 nM T56418 C1MF0Z 56650031 IC50 = 1 nM T56418 C9E2UL 56650032 IC50 = 2 nM T56418 CTF2M1 56650355 IC50 = 1 nM T56418 CF45NV 56650693 IC50 = 109 nM T56418 C3A0YT 56650694 IC50 = 1.6 nM T56418 C59XFV 56653076 IC50 = 1 nM T56418 CM1LX6 56653440 IC50 = 44 nM T56418 CR75VU 56653441 IC50 = 5 nM T56418 C0T5AY 56653442 IC50 = 24 nM T56418 CW20UD 56654475 IC50 = 2 nM T56418 C5FNZ4 56654813 IC50 = 13 nM T56418 CV81ZS 56654815 IC50 = 1.5 nM T56418 CIY0W9 56654816 IC50 = 1.6 nM T56418 C8WH7U 56655160 IC50 = 2 nM T56418 CQOU10 56655161 IC50 = 2 nM T56418 CBZ8T4 56657856 IC50 = 2375 nM T56418 CGZ76M 56658177 IC50 = 8.8 nM T56418 C9RO7H 56659710 IC50 = 65 nM T56418 CQX1B0 56659754 IC50 > 40000 nM T56418 CPEQ43 56659755 IC50 > 40000 nM T56418 CM15EG 56659756 IC50 > 40000 nM T56418 COT59W 56659757 IC50 > 40000 nM T56418 C9JN5I 56659776 IC50 > 40000 nM T56418 CO6XJ2 56659777 IC50 > 40000 nM T56418 CO7N3J 56659778 IC50 = 7540 nM T56418 CR2AZ4 56659779 IC50 > 40000 nM T56418 CP02ZN 56663035 IC50 = 9000 nM T56418 C0TA4N 56663131 IC50 > 40000 nM T56418 C10HLV 56663132 IC50 > 40000 nM T56418 C8CRO9 56663133 IC50 > 40000 nM T56418 CVL35R 56663134 IC50 > 40000 nM T56418 C4AJE2 56663169 IC50 = 330 nM T56418 C3ZXK9 56663170 IC50 > 10000 nM T56418 C3R4VA 56663171 IC50 = 200 nM T56418 C28VGO 56663172 IC50 = 22 nM T56418 CQ9RN5 56663173 IC50 = 680 nM T56418 C0BKE4 56663174 IC50 = 150 nM T56418 CQLP34 56663175 IC50 > 3000 nM T56418 CC6Y5B 56663231 IC50 > 40000 nM T56418 CTPK64 56663250 IC50 > 40000 nM T56418 CWYO21 56663251 IC50 = 6910 nM T56418 CFMW78 56663252 IC50 > 40000 nM T56418 CP07FJ 56665099 IC50 = 9 nM T56418 C0NCP7 56666587 IC50 > 40000 nM T56418 C8XZ4O 56666620 IC50 = 300 nM T56418 CZDJ40 56666621 IC50 = 110 nM T56418 CML6O1 56666622 IC50 > 3000 nM T56418 CI9CK1 56666661 IC50 > 40000 nM T56418 CKBD90 56666683 IC50 > 40000 nM T56418 C0Q4XE 56666684 IC50 > 40000 nM T56418 CEH31Y 56668417 IC50 = 212 nM T56418 CI4GQ9 56670029 IC50 = 100 nM T56418 C9DJH8 56670079 IC50 > 40000 nM T56418 C46PYQ 56670080 IC50 > 40000 nM T56418 C37WLX 56670081 IC50 > 40000 nM T56418 CB83JE 56670082 IC50 > 40000 nM T56418 C8A4RP 56670104 IC50 > 40000 nM T56418 CC54FO 56670105 IC50 > 40000 nM T56418 C01WYS 56673544 IC50 > 3000 nM T56418 C9OA3E 56673602 IC50 > 40000 nM T56418 C59WKG 56673603 IC50 > 40000 nM T56418 C4HKA0 56673622 IC50 > 40000 nM T56418 C9TH6I 56673623 IC50 = 6250 nM T56418 CYPL60 56675140 IC50 > 10000 nM T56418 CSZ9P6 56676866 IC50 = 10 nM T56418 CMO45E 56676867 IC50 = 9 nM T56418 CLMK58 56676868 IC50 = 50 nM T56418 C07DET 56676869 IC50 = 15 nM T56418 CFC14P 56676919 IC50 > 40000 nM T56418 CXQ3W5 56676939 IC50 > 40000 nM T56418 CS92FR 56676940 IC50 > 40000 nM T56418 C87OYI 56676941 IC50 > 40000 nM T56418 C4RJ5H 56680184 IC50 = 60 nM T56418 C8GT6K 56680185 IC50 = 78 nM T56418 C4ARS6 56680232 IC50 > 40000 nM T56418 C7XH1J 56680233 IC50 > 40000 nM T56418 CE8N6R 56680259 IC50 = 6640 nM T56418 CO21ZG 56680260 IC50 = 7570 nM T56418 C86EIX 56680261 IC50 = 7540 nM T56418 C45RZV 56683336 IC50 = 370 nM T56418 CN5W3I 56683485 IC50 > 40000 nM T56418 CE84TZ 56683526 IC50 = 130 nM T56418 C8ZJE5 56683588 IC50 = 10180 nM T56418 C5UKI1 56683589 IC50 > 40000 nM T56418 C7Y2EO 56683590 IC50 = 9870 nM T56418 CA09TN 56945204 IC50 = 22 nM T56418 CCDG27 56945394 IC50 = 56 nM T56418 C9VK2H 56945491 IC50 = 14 nM T56418 C5F8CI 56945493 IC50 = 6 nM T56418 C1AE3J 56945494 IC50 = 6 nM T56418 CL4AS8 56945495 IC50 = 10 nM T56418 C60HVN 56945611 IC50 = 3.4 nM T56418 CN1A8C 56945612 IC50 = 6 nM T56418 CGW9B2 56945613 IC50 = 3 nM T56418 CE95CG 56945614 IC50 = 2.9 nM T56418 CA3U2R 56945615 IC50 = 7 nM T56418 C6AJC0 56945727 IC50 = 10 nM T56418 C5FY9U 56945728 IC50 = 6 nM T56418 C2OS1K 56945729 IC50 = 12 nM T56418 CWS36I 56945730 IC50 = 19 nM T56418 CY39NF 56945731 IC50 = 1061 nM T56418 CNS43L 56945844 IC50 = 9 nM T56418 CF0X2H 56945845 IC50 = 15 nM T56418 C79TMP 56945846 IC50 = 6 nM T56418 C9VA7E 56945847 IC50 = 4.7 nM T56418 CG43UB 56946521 IC50 = 67 nM T56418 CZ87NL 56946522 IC50 > 10000 nM T56418 CC4L3K 56946524 IC50 = 283 nM T56418 CA6BT1 56946619 IC50 = 92 nM T56418 CH9M0Y 56946621 IC50 > 1000 nM T56418 C6BH3W 56946623 IC50 = 150 nM T56418 CL8WZ3 56946626 IC50 = 3.7 nM T56418 C7RFK3 56946730 IC50 = 120 nM T56418 CBZJ82 56946732 IC50 = 800 nM T56418 CO6HY1 56946734 IC50 = 30 nM T56418 C6F9VJ 56946736 IC50 = 0.51 nM T56418 CF5JV6 56966833 IC50 = 0.18 nM T56418 C1WJT2 56966906 IC50 = 1.03 nM T56418 C26MCX 56966977 IC50 = 0.76 nM T56418 CX34KP 56966978 IC50 = 0.38 nM T56418 C56XYJ 57325607 IC50 = 95 nM T56418 C09DJP 57325609 IC50 = 70 nM T56418 C95OSR 57325611 IC50 = 2930 nM T56418 CJ93CQ 57325613 IC50 = 60 nM T56418 CB6UG1 57325697 IC50 = 1700 nM T56418 CZUV79 57325700 IC50 = 138 nM T56418 CKQF98 57325702 IC50 = 192 nM T56418 CGN9R7 57326499 IC50 = 4120 nM T56418 C1M2SJ 57326501 IC50 > 25000 nM T56418 C7HSP3 57326503 IC50 = 2320 nM T56418 C06SPM 57326505 IC50 > 25000 nM T56418 CIRD14 57326601 IC50 = 2010 nM T56418 CUCT15 57326603 IC50 = 6300 nM T56418 CY5AW1 57326605 IC50 = 1020 nM T56418 CY6JT2 57326607 IC50 = 3100 nM T56418 C8X0KC 57326609 IC50 = 912 nM T56418 CNW2D1 57326700 IC50 > 25000 nM T56418 CSV93R 57326702 IC50 = 1730 nM T56418 C0QU2R 57326704 IC50 = 1480 nM T56418 CML95J 57326706 IC50 = 325 nM T56418 CF65OP 57326708 IC50 = 833 nM T56418 C5K1TC 57326800 IC50 = 364 nM T56418 C1Y9WO 57326802 IC50 = 358 nM T56418 C5P8CS 57326804 IC50 = 6710 nM T56418 CH92NG 57326806 IC50 = 2940 nM T56418 CIE2N9 57326900 IC50 = 2600 nM T56418 CT4HO0 57326902 IC50 = 2010 nM T56418 C6DWX9 57326904 IC50 = 341 nM T56418 C86FYD 57326906 IC50 = 83 nM T56418 CU8L3K 57326995 IC50 = 587 nM T56418 C4AI8K 57326997 IC50 = 80 nM T56418 CDW6R2 57329726 IC50 = 1 nM T56418 CW8A0C 57345939 IC50 = 5 nM T56418 CWM1B3 57345940 IC50 = 3 nM T56418 CN96HJ 57392673 IC50 = 229 nM T56418 CE8T5V 57393795 IC50 > 20000 nM T56418 CMG03J 57394376 IC50 = 63 nM T56418 C3VNY5 57394377 IC50 = 100 nM T56418 C3UHX0 57394704 IC50 = 69.3 nM T56418 CD0OQ4 57396144 IC50 = 46 nM T56418 CE1WT0 57396145 IC50 = 13 nM T56418 CD7C4R 57396463 IC50 = 16 nM T56418 C03CUD 57397961 IC50 = 104 nM T56418 C9BUV4 57397962 IC50 = 120 nM T56418 C6HJ1A 57397963 IC50 = 42 nM T56418 CS51TX 57398770 IC50 = 35 nM T56418 C4Y0BJ 57399599 IC50 = 54 nM T56418 CX2UW6 57399904 IC50 = 233 nM T56418 CE31FR 57399905 IC50 = 5.2 nM T56418 C7VN0E 57401361 IC50 = 10000 nM T56418 C3E4MA 57401677 IC50 = 44 nM T56418 CK06MA 57402935 IC50 = 30 nM T56418 CGE8I2 57403115 IC50 = 46 nM T56418 C7T0CM 57403116 IC50 = 4600 nM T56418 C16GQE 57403117 IC50 = 17 nM T56418 CP9Z4O 57403409 IC50 = 67 nM T56418 CRU80Y 57403410 IC50 = 1.1 nM T56418 C08CUY 57522736 IC50 = 21 nM T56418 CZ6I9Y 57522737 IC50 = 9 nM T56418 CPL2K0 57522850 IC50 = 35 nM T56418 CL12XK 58009759 IC50 = 380 nM T56418 CTWG72 58290872 IC50 = 25.8 nM T56418 C24BEZ 59577331 IC50 = 15 nM T56418 C1JCV8 59577340 IC50 = 181 nM T56418 CT3J2N 59577341 IC50 = 67 nM T56418 C1CSH0 59577345 IC50 = 99 nM T56418 CJZ71Q 59577355 IC50 = 26 nM T56418 CIB62O 59577356 IC50 = 18 nM T56418 C75VNB 59577361 IC50 = 106 nM T56418 C7QY2B 59577365 IC50 = 9 nM T56418 CPU2E3 59737752 IC50 = 24.8 nM T56418 CF8E1J 59764390 IC50 = 36.4 nM T56418 CC48EN 59764418 IC50 = 10.6 nM T56418 C4NBG7 59764433 IC50 = 17.3 nM T56418 C40UZT 59764460 IC50 = 8.1 nM T56418 C6AQX8 59764524 IC50 = 11.5 nM T56418 C5B0JN 59764577 IC50 = 258.4 nM T56418 CRZ9M5 60195567 IC50 = 2 nM T56418 C6BTI1 60195647 IC50 = 7 nM T56418 C7A0SD 60195648 IC50 = 1.6 nM T56418 CO7K1T 60195649 IC50 = 1.2 nM T56418 CNQC96 60195650 IC50 = 144 nM T56418 C8BGT2 60195732 IC50 = 2 nM T56418 C84BHI 60195733 IC50 = 1.4 nM T56418 CBU76J 60195734 IC50 = 2 nM T56418 CCB3G0 60195735 IC50 = 8 nM T56418 CQR7H2 60195826 IC50 = 2 nM T56418 C0N2DV 60195911 IC50 = 1 nM T56418 CHE17Z 60195912 IC50 = 1 nM T56418 CD24TN 60195913 IC50 = 6 nM T56418 C14IBA 60195914 IC50 = 3 nM T56418 CCY8P6 60195999 IC50 = 3 nM T56418 CXR75J 60196000 IC50 = 2 nM T56418 C6B7AD 60196001 IC50 = 3 nM T56418 C3E7OI 60196002 IC50 = 1 nM T56418 C08VMZ 60198892 IC50 = 177 nM T56418 C9ZCT2 62705065 IC50 = 348.9 nM T56418 C8KB9Q 66710864 IC50 = 15 nM T56418 CZU92Y 66711083 IC50 = 3 nM T56418 CBD83S 66711091 IC50 = 6 nM T56418 C3FA7X 66711377 IC50 = 3 nM T56418 C1P0LG 66711384 IC50 = 8 nM T56418 CEXY72 66711391 IC50 = 3 nM T56418 CZGJ30 66711499 IC50 = 15 nM T56418 CHN8T6 66711835 IC50 = 57 nM T56418 CNC0V3 66711879 IC50 = 40 nM T56418 CY0C3J 66829998 IC50 = 39 nM T56418 C82YDV 66830004 IC50 = 11 nM T56418 CMN68E 66830116 IC50 = 30 nM T56418 CX7LS6 66830288 IC50 = 8 nM T56418 CY31IS 66830367 IC50 = 2139 nM T56418 COH5N4 66830485 IC50 = 5 nM T56418 CBU5X6 66830555 IC50 = 568 nM T56418 CRH43K 66830651 IC50 = 4 nM T56418 C2HRJ9 66830713 IC50 = 3200 nM T56418 C1HSE0 67035086 IC50 = 760 nM T56418 CWI6K5 67035106 IC50 > 10000 nM T56418 C38RGB 67035556 IC50 > 10000 nM T56418 C37NKO 67129970 IC50 = 7630 nM T56418 CK80LJ 67130050 IC50 = 5940 nM T56418 CV63UL 67240318 IC50 > 10000 nM T56418 CI9P5C 67263749 IC50 = 6 nM T56418 C0F1UO 67263935 IC50 = 4 nM T56418 CDE47U 67264047 IC50 = 7 nM T56418 CI41EV 67264228 IC50 = 15 nM T56418 C9YIN0 67264246 IC50 = 3.1 nM T56418 C7BF3N 67264510 IC50 = 40 nM T56418 C7XU0T 67425014 IC50 = 60 nM T56418 C1K3TA 67462112 Ki = 2.6 nM T56418 C0HM1N 67467673 Ki = 7.5 nM T56418 CQCN08 67467779 Ki = 4 nM T56418 CEV60X 68156947 IC50 = 0.31 nM T56418 C59RQC 68165302 IC50 = 0.12 nM T56418 CL97JB 68165311 IC50 = 0.24 nM T56418 CM1ZC3 68165315 IC50 = 0.22 nM T56418 CET2P8 68165322 IC50 = 0.28 nM T56418 C61QGN 68165327 IC50 = 0.33 nM T56418 CFRK82 68165328 IC50 = 0.33 nM T56418 CLH97K 68165338 IC50 = 0.39 nM T56418 C7Y8KG 68165350 IC50 = 0.36 nM T56418 C2AX3V 68165354 IC50 = 0.49 nM T56418 C2B3TL 68165357 IC50 = 0.42 nM T56418 C81YOZ 68165362 IC50 = 0.54 nM T56418 CLGN08 68165375 IC50 = 0.68 nM T56418 C82RIW 68165380 IC50 = 0.75 nM T56418 CH5Y2P 68165382 IC50 = 0.72 nM T56418 C3H5XQ 68165389 IC50 = 0.88 nM T56418 C0WFX2 68165395 IC50 = 0.79 nM T56418 C0G7QF 68165398 IC50 = 0.68 nM T56418 CNK7S3 68165399 IC50 = 0.59 nM T56418 C78BZG 68165403 IC50 = 0.53 nM T56418 CZ1Q8W 68165412 IC50 = 0.96 nM T56418 CYD2V8 68165414 IC50 = 0.86 nM T56418 CVGJ74 68165424 IC50 = 1.36 nM T56418 C9NA2W 68165441 IC50 = 2.1 nM T56418 CN27QC 68165467 IC50 = 3.23 nM T56418 CO2LF9 68166178 IC50 = 0.88 nM T56418 CR1U7L 68166323 IC50 = 0.33 nM T56418 C4VQJ8 68166330 IC50 = 3.1 nM T56418 C8I7GC 68293638 IC50 > 10000 nM T56418 CD56XK 68293660 IC50 > 10000 nM T56418 C7GRV2 68755406 IC50 > 10000 nM T56418 CAI3J4 70654537 IC50 > 10000 nM T56418 C7F4DB 70654775 IC50 = 4500 nM T56418 CA0UR2 70654830 IC50 = 860 nM T56418 C49KEL 70655062 IC50 = 559 nM T56418 CXU06B 70660512 IC50 = 1200 nM T56418 CTJ6D0 70661442 IC50 = 5642 nM T56418 CV6TZ8 70661443 IC50 = 805 nM T56418 CC90HU 70684001 IC50 = 1000 nM T56418 CB1X4E 70696546 IC50 = 100 nM T56418 C3ZB4V 71451378 IC50 = 187 nM T56418 C1GN3W 71458548 IC50 = 28 nM T56418 C7LCS8 71470563 IC50 = 40 nM T56418 C9DIK2 71512060 IC50 > 10000 nM T56418 CCN01X 71547862 IC50 > 10000 nM T56418 CW4NI7 71604335 IC50 = 29 nM T56418 C3OS8U 71714087 IC50 = 370 nM T56418 C92AZQ 71714088 IC50 = 1500 nM T56418 CN1Y9I 71714230 IC50 = 1400 nM T56418 CM6NE9 71714231 IC50 = 550 nM T56418 CG28AP 71714232 IC50 = 660 nM T56418 C91CRY 71714233 IC50 > 10000 nM T56418 C67HDT 71714234 IC50 > 10000 nM T56418 CRS05F 71714235 IC50 = 76 nM T56418 CVC19T 71714373 IC50 = 210 nM T56418 CD5C8J 71714374 IC50 = 3300 nM T56418 C51ISR 71714375 IC50 = 9500 nM T56418 C5HJK2 71714376 IC50 = 1600 nM T56418 C70SJV 71714377 IC50 > 10000 nM T56418 CYS9Q0 71731827 Ki < 0.2 nM T56418 CX9DI8 71732092 Ki = 0.38 nM T56418 C5DV0R 71732094 Ki < 0.1 nM T56418 CP1LE8 71732095 Ki = 0.36 nM T56418 C2F3DA 71732097 Ki = 5 nM T56418 C72KYC 71763639 IC50 = 48.3 nM T56418 C8ZY1V 71763864 IC50 = 4240 nM T56418 C19WUN 71764054 IC50 = 40.6 nM T56418 C56IPY 71764055 IC50 = 38.1 nM T56418 CG5S3Y 71764056 IC50 = 32.1 nM T56418 CS8BR1 71764218 IC50 = 29.9 nM T56418 CNW35A 71764219 IC50 = 305.7 nM T56418 CS6DN3 71764394 IC50 = 88.9 nM T56418 CUGC68 71764395 IC50 = 16.5 nM T56418 C2NJ4Z 71764396 IC50 = 29.4 nM T56418 CGWT31 71764397 IC50 = 63.6 nM T56418 C0KNW2 71764604 IC50 = 44 nM T56418 CMI76L 71818269 IC50 = 85 nM T56418 C6UJ9Z 71818270 IC50 = 35 nM T56418 CCN4Q0 71818271 IC50 = 70 nM T56418 CNID49 71818272 IC50 = 30 nM T56418 CIS29B 71818419 IC50 = 32 nM T56418 CTO83G 71818420 IC50 = 247 nM T56418 CVJ2I0 71818421 IC50 = 98 nM T56418 CN06TE 71818422 IC50 = 70 nM T56418 C8C7KM 71818423 IC50 = 28 nM T56418 CR98AM 71818424 IC50 = 41 nM T56418 CRKF01 71818562 IC50 = 985.6 nM T56418 CY9RP8 71818563 IC50 = 6 nM T56418 C6W9BO 71818564 IC50 = 56 nM T56418 C4I0BA 71818565 IC50 = 31 nM T56418 C0VS6U 71818566 IC50 = 63 nM T56418 C7J9ZQ 71818703 IC50 = 310.2 nM T56418 CB64IQ 72194525 IC50 = 94.1 nM T56418 C1OCE8 73057484 IC50 = 90 nM T56418 CZN1Y6 73354960 IC50 > 10000 nM T56418 CVNW01 73386831 IC50 > 1000 nM T56418 C45BPD 73819542 Ki = 0.85 nM T56418 CYK09C 73819543 Ki < 0.2 nM T56418 CRI51K 73819548 Ki < 0.1 nM T56418 C3UC9H 73891099 IC50 = 180 nM T56418 C3E9MB 76281906 IC50 = 15 nM T56418 CAZ5N3 76281907 IC50 = 3.5 nM T56418 CTKJ62 76281908 IC50 = 14 nM T56418 C19PGZ 76282166 IC50 = 50 nM T56418 CTEF85 76282167 IC50 = 60 nM T56418 CC2K0H 76282402 IC50 > 1000 nM T56418 CEW67B 76282644 IC50 = 38 nM T56418 CV8QX0 76310169 IC50 = 9760 nM T56418 CDBJ72 76310629 IC50 = 49000 nM T56418 C67DFL 76311143 Ki = 6.1 nM T56418 CAM0H5 76311144 Ki < 0.2 nM T56418 CIBN36 76314256 IC50 = 51000 nM T56418 CC6I8K 76314257 IC50 = 3500 nM T56418 C8E4IL 76314258 IC50 = 1500 nM T56418 CQ2SA5 76317829 IC50 = 52000 nM T56418 C28YHN 76317830 IC50 = 2200 nM T56418 C3M1NA 76318349 Ki = 9 nM T56418 C13NZF 76318350 Ki = 15 nM T56418 CB9XW7 76321540 IC50 = 10000 nM T56418 C25JOE 76321541 IC50 > 100000 nM T56418 CU3LB2 76322031 Ki = 2.8 nM T56418 CXN2V3 76322032 Ki = 1.3 nM T56418 C74CNR 76322033 Ki = 190 nM T56418 CEB13H 76322034 Ki = 5 nM T56418 CA5L4W 76324771 IC50 = 9330 nM T56418 CAE07Q 76325144 IC50 > 100000 nM T56418 C7GNS8 76325654 Ki = 0.6 nM T56418 C81DZC 76325655 Ki = 2.6 nM T56418 C9GO0P 76328313 IC50 = 5020 nM T56418 C3JDO5 76328703 IC50 = 9000 nM T56418 C1B2JP 76329225 Ki = 1.1 nM T56418 CS0YD1 76332386 IC50 > 50000 nM T56418 C6N7IP 76332387 IC50 = 29000 nM T56418 C16ADY 76332388 IC50 = 14000 nM T56418 CIU90K 76332880 Ki = 0.3 nM T56418 C6GT8C 76332881 Ki = 16 nM T56418 CY57OB 76332882 Ki = 2 nM T56418 CJ2T9E 76332983 IC50 = 2200 nM T56418 C39FTZ 76335685 IC50 = 3380 nM T56418 CR6EK4 76336015 IC50 = 18000 nM T56418 C3OS1F 76336490 Ki = 11 nM T56418 CH8W7D 77461036 IC50 = 2.7 nM T56418 CQZ0L8 78158242 IC50 = 3.4 nM T56418 CH3FN8 86288905 IC50 = 5 nM T56418 CBGN34 86292464 IC50 = 63.42 nM T56418 CPG3A5 86302574 IC50 > 30000 nM T56418 CQU3C5 89713230 Ki < 0.2 nM T56418 C58VLT 89726147 IC50 = 29 nM T56418 CA49UY 89726151 IC50 = 0.76 nM T56418 CY6K5P 89738540 IC50 = 60 nM T56418 CIXB02 89738547 IC50 = 0.31 nM T56418 CH58TV 89773144 IC50 = 1.19 nM T56418 CSX63K 89773146 IC50 = 1.88 nM T56418 CTV2C7 89774514 IC50 = 0.49 nM T56418 C6R2TS 89807790 Ki = 0.1 nM T56418 CXV69E 89808089 Ki = 4 nM T56418 CAQE21 89808124 Ki < 0.07 nM T56418 CRSY98 89808125 Ki = 2 nM T56418 C40VNJ 89816720 Ki = 0.56 nM T56418 CFB75T 90479825 IC50 = 143 nM T56418 CM64AB 90644193 Ki < 0.2 nM T56418 CMP9N8 90644194 Ki = 2.8 nM T56418 CV73MS 90644195 Ki = 22 nM T56418 C3FRG0 90644196 Ki < 0.1 nM T56418 CNLQ51 90644197 Ki < 0.1 nM T56418 CI9T6Z 90644198 Ki = 17 nM T56418 C1B4AZ 90644199 Ki = 0.1 nM T56418 C8G4JY 90644200 Ki = 17 nM T56418 CM8NY2 90644201 Ki < 0.02 nM T56418 CA0T8V 90644202 Ki < 0.1 nM T56418 CY0UC4 90645194 IC50 > 10000 nM T56418 CHAQ83 90655778 IC50 = 7.7 nM T56418 CNB2K3 90655779 IC50 = 19 nM T56418 C3TM0S 90655780 IC50 = 17 nM T56418 C6V7KD 90655781 IC50 = 13 nM T56418 C7TS4O 90655782 IC50 = 17 nM T56418 CPW01E 90655783 IC50 = 36 nM T56418 C1G6QK 90655784 IC50 = 7.9 nM T56418 CV1S6R 90655785 IC50 = 53 nM T56418 CDWP34 90655786 IC50 > 1000 nM T56418 CKD16A 90655787 IC50 > 1000 nM T56418 C6EUD2 90655788 IC50 > 1000 nM T56418 CO28UJ 90655789 IC50 > 1000 nM T56418 CAU5K7 90655790 IC50 > 1000 nM T56418 C5NZ7A 90655791 IC50 > 1000 nM T56418 CGP7R9 90655792 IC50 = 7.1 nM T56418 C42VGQ 90655793 IC50 = 1.3 nM T56418 CM38BR 90655794 IC50 = 49 nM T56418 C4GU0L 90665978 IC50 = 199 nM T56418 CP65IG 90665979 IC50 = 212 nM T56418 CZA0F4 90665980 IC50 = 16 nM T56418 CJF1Z9 90665981 IC50 = 85 nM T56418 CY90XF 90665982 IC50 = 121 nM T56418 CR1Q9I 90665983 IC50 = 4 nM T56418 CV62FB 90665984 IC50 = 270 nM T56418 C8EUC3 90665985 IC50 = 42 nM T56418 CXEJ32 90665986 IC50 = 7 nM T56418 CDQ56W 90665987 IC50 = 0.69 nM T56418 C5E2FJ 90665988 IC50 = 8 nM T56418 C4TPN8 90665989 IC50 = 2.7 nM T56418 CP59DM 90665990 IC50 > 10000 nM T56418 C10HSM 90665991 IC50 > 3000 nM T56418 CBG6E7 91885506 IC50 = 5.7 nM T56418 C3N5IY 117955447 IC50 = 2 nM T56418 C4CH7J 117955548 IC50 = 4 nM T56418 C5T4WU 117955577 IC50 = 2.3 nM T56418 C2T4MB 117955613 IC50 = 44 nM T56418 C07ACT 117955744 IC50 = 2.3 nM T56418 C5K2DA 117955863 IC50 = 5 nM T56418 C50ANY 117955890 IC50 = 18 nM T56418 CTOY69 118549502 IC50 = 8 nM T56418 CC7NG2 118549504 IC50 = 8 nM T56418 CRA9N7 118549506 IC50 = 5 nM T56418 CM7JP2 118549507 IC50 = 7 nM T56418 CV1EX5 118549510 IC50 = 2 nM T56418 CG1J5R 118549511 IC50 = 3 nM T56418 CL1BC5 118549519 IC50 = 1 nM T56418 C8V6YN 118549529 IC50 = 3 nM T56418 CL0G1P 118549537 IC50 = 2 nM T56418 C21OHF 118549540 IC50 = 22 nM T56418 CL0Y3U 118549545 IC50 = 16 nM T56418 CUK4I2 118549558 IC50 = 2 nM T56418 CLO7U0 118549683 IC50 = 4 nM T56418 C09RMO 118549795 IC50 = 6 nM T56418 CP9E4B 118549812 IC50 = 12 nM T56418 C5VS6A 118549813 IC50 = 23 nM T56418 CWHA28 118549821 IC50 = 22 nM T56418 CMH53T 118549960 IC50 = 16 nM T56418 CW7ZX4 118550024 IC50 = 3 nM T56418 CY7BI2 118706214 IC50 > 10000 nM T56418 CI28QB 118713249 IC50 = 61.8 nM T56418 C7S6BN 118713250 IC50 > 1000000 nM T56418 CAQL94 118713251 IC50 = 99 nM T56418 CN27MB 118713252 IC50 = 773 nM T56418 C8OX0R 118713253 IC50 = 171 nM T56418 C47XYM 118713254 IC50 = 178 nM T56418 CW3VE2 118713255 IC50 > 1000000 nM T56418 C0ASF3 118713256 IC50 > 1000000 nM T56418 CYUR03 118713257 IC50 = 18 nM T56418 C37ECP 118713258 IC50 = 24 nM T56418 CU4SF1 118713259 IC50 = 67.8 nM T56418 CD75UM 118713260 IC50 > 1000 nM T56418 CZ4TU2 118713261 IC50 > 1000 nM T56418 CMP7X0 118713262 IC50 = 775 nM T56418 CGZ35A 118713263 IC50 > 1000 nM T56418 C0ALV5 118713264 IC50 > 1000 nM T56418 C0O2HX 118713265 IC50 > 1000 nM T56418 CQ8K1S 118713266 IC50 > 1000 nM T56418 CPB21W 118713267 IC50 > 1000 nM T56418 C7HXT3 118713268 IC50 = 121 nM T56418 C2PEY3 118713269 IC50 > 1000 nM T56418 CN7R4V 118713270 IC50 = 471 nM T56418 C6FSM1 118713271 IC50 > 1000 nM T56418 CQ81EM 118713272 IC50 > 1000 nM T56418 C1J2IC 118713273 IC50 = 144 nM T56418 CW05OQ 118713274 IC50 > 1000 nM T56418 CM1QS8 118713275 IC50 = 134 nM T56418 CYPK49 118713276 IC50 = 243 nM T56418 CYLJ17 118713277 IC50 > 1000 nM T56418 C0IUS3 118721850 IC50 = 32.8 nM T56418 C1NZT3 118721851 IC50 > 1000 nM T56418 C9IR6M 118721852 IC50 = 280 nM T56418 CA07OH 118722207 IC50 = 80.3 nM T56418 CZ93GF 118722208 IC50 > 1000 nM T56418 CKM9F5 118722209 IC50 = 111 nM T56418 CJU8I4 118722210 IC50 = 94.5 nM T56418 CBXC83 118722211 IC50 = 7.7 nM T56418 C9JMP7 118722212 IC50 > 1000 nM T56418 C4IG8N 118722213 IC50 = 1.8 nM T56418 CM9B4L 118722214 IC50 = 14.9 nM T56418 CW3HP9 118722215 IC50 = 50.8 nM T56418 COI93D 118722216 IC50 = 5.5 nM T56418 CFN94B 118722217 IC50 = 28 nM T56418 CHX3I0 118722218 IC50 = 3.1 nM T56418 C8TBS4 118722219 IC50 = 19.1 nM T56418 C8Q6ON 118722220 IC50 = 44.2 nM T56418 CB7G8S 118722221 IC50 = 20.7 nM T56418 CTWA53 118722222 IC50 = 0.8 nM T56418 C3BLR8 118722223 IC50 = 17.8 nM T56418 CWTY65 118722224 IC50 = 25.5 nM T56418 C1ROT4 118722225 IC50 = 2.5 nM T56418 CIC5R2 118722226 IC50 = 1.7 nM T56418 C8UTX5 118722227 IC50 = 4.9 nM T56418 CY9W0C 118722228 IC50 = 0.7 nM T56418 CU8KS3 118722229 IC50 = 9 nM T56418 CVC74S 118722230 IC50 = 2.3 nM T56418 C5WR9T 118722231 IC50 = 51.3 nM T56418 CO9CG3 118722232 IC50 = 3 nM T56418 CEFM78 118722233 IC50 = 2.3 nM T56418 C9OXS4 118722234 IC50 = 5.5 nM T56418 C2Z3FV 118722235 IC50 = 31.9 nM T56418 CHQ19T 118722236 IC50 = 95.3 nM T56418 CW4O3Q 118726562 IC50 = 4320 nM T56418 CO8YT9 118726563 IC50 = 1920 nM T56418 C3CSO5 118726564 IC50 = 10200 nM T56418 C9PW5V 118726565 IC50 = 6220 nM T56418 CI50GB 118726567 IC50 = 9720 nM T56418 CW7U2O 118726568 IC50 = 4150 nM T56418 CCK37S 118726569 IC50 = 20000 nM T56418 C5PX2O 118726570 IC50 = 17600 nM T56418 C0VK2L 118988436 IC50 = 4 nM T56418 CBPN57 119025617 IC50 = 402 nM T56418 CU3AW9 119025618 IC50 > 10000 nM T56418 C08KEM 122179540 IC50 = 3100 nM T56418 C3AJ4C 122179546 IC50 = 6300 nM T56418 CG0RP7 122179547 IC50 = 1200 nM T56418 C1A0SQ 122179548 IC50 = 3900 nM T56418 C7FD4R 122185893 IC50 = 1 nM T56418 CW2Q7M 122185894 IC50 = 10 nM T56418 CVK83H 122185895 IC50 = 15 nM T56418 C1X7GL 122185896 IC50 = 3 nM T56418 CEW25Z 122185897 IC50 = 4 nM T56418 CNK4A0 122185898 IC50 = 4 nM T56418 C46DHF 122185899 IC50 = 13 nM T56418 C0SJX4 122185900 IC50 = 4 nM T56418 C3INE4 122185901 IC50 = 5 nM T56418 CE98GO 122185902 IC50 = 5 nM T56418 C2TGQ9 122185903 IC50 = 7 nM T56418 CIO8F2 122185904 IC50 = 4 nM T56418 C9C3PS 122185905 IC50 = 10 nM T56418 CR9UY2 122185906 IC50 = 2 nM T56418 CX4A6F 122185907 IC50 = 26 nM T56418 C4OG2Y 122185908 IC50 = 9 nM T56418 CRX5O8 122185909 IC50 = 6 nM T56418 CND7S8 122186934 IC50 = 3 nM T56418 CUBD36 122186935 IC50 = 4.4 nM T56418 CP65NK 122186936 IC50 = 15 nM T56418 CA74DF 122186937 IC50 = 1.7 nM T56418 CK8G1M 122186938 IC50 = 1.6 nM T56418 CCR3P8 122186939 IC50 = 1.8 nM T56418 CQW9Z5 122186940 IC50 = 1.5 nM T56418 CF4YM1 122186941 IC50 = 1400 nM T56418 C2K6TV 122186942 IC50 = 2000 nM T56418 C0J2PX 122186943 IC50 = 1000 nM T56418 CRP30D 122186944 IC50 = 2700 nM T56418 C78ELB 122186945 IC50 = 800 nM T56418 CSV10H 122186946 IC50 = 1000 nM T56418 CH9OX7 122186947 IC50 = 4500 nM T56418 CWP9Z4 122186948 IC50 = 2100 nM T56418 C6G9PD 122186949 IC50 = 600 nM T56418 CI9EW1 122186950 IC50 = 35000 nM T56418 CB1I7P 122187040 IC50 = 700 nM T56418 C19SRK 122187041 IC50 = 2500 nM T56418 C8VA2S 122187042 IC50 = 1200 nM T56418 CC5WV2 122187043 IC50 = 7300 nM T56418 C57NJT 122187044 IC50 = 2400 nM T56418 CJ9EN3 122187045 IC50 = 3400 nM T56418 C24AKR 122187525 IC50 = 1700 nM T56418 CD54PM 126747042 IC50 = 8 nM T56418 CVY92K 126747046 IC50 = 7 nM T56418 CQE7W4 126747054 IC50 = 6 nM T56418 CBH32U 126747059 IC50 = 9 nM T56418 C62OWQ 127030997 IC50 = 29 nM T56418 CQ0R4I 127030998 IC50 = 18 nM T56418 CH93CT 127030999 IC50 = 8.4 nM T56418 C7KZN9 127031000 IC50 = 40 nM T56418 CV0NK3 127031324 IC50 = 27 nM T56418 C2V5GI 127031588 IC50 = 342 nM T56418 C2UNF0 127031589 IC50 = 43 nM T56418 CV72PY 127031598 IC50 = 16 nM T56418 CZ2KR8 127031879 IC50 = 56 nM T56418 C2Z0DY 127031880 IC50 = 424 nM T56418 C1ZSX0 127031881 IC50 = 52 nM T56418 CFO87C 127031882 IC50 = 44 nM T56418 CFS98V 127031883 IC50 = 122 nM T56418 CM4R0X 127031884 IC50 = 212 nM T56418 C2YTW3 127031885 IC50 = 21 nM T56418 CR9HZ5 127032117 IC50 = 34 nM T56418 CYHK91 127032122 IC50 = 1.5 nM T56418 C16GKO 127032123 IC50 = 9.9 nM T56418 CJ6M9L 127032124 IC50 = 3.6 nM T56418 CMXI71 127032144 IC50 = 16 nM T56418 CUV61A 127032214 IC50 = 3 nM T56418 C5VNR7 127032501 IC50 = 20 nM T56418 CI7FQ5 127032502 IC50 = 129 nM T56418 C43SJK 127032810 IC50 = 400 nM T56418 CJV0T3 127032811 IC50 = 6683 nM T56418 C21TER 127032812 IC50 = 12 nM T56418 CD6GE1 127033964 IC50 = 22 nM T56418 CD9XL1 127033965 IC50 = 56 nM T56418 C9QS4D 127034224 IC50 = 753 nM T56418 CU2E6I 127034492 IC50 = 36 nM T56418 CR07QN 127034799 IC50 = 2.1 nM T56418 C10MJV 127034800 IC50 = 2.3 nM T56418 CSDF05 127034801 IC50 = 15.5 nM T56418 CKS28E 127034802 IC50 = 3.4 nM T56418 C8R7CD 127034822 IC50 = 5.6 nM T56418 CGI2B5 127035975 IC50 = 4.1 nM T56418 C5AL9F 127035976 IC50 = 0.8 nM T56418 CRL51P 127035977 IC50 = 2.1 nM T56418 CE2Z1I 127036114 IC50 = 23 nM T56418 CBA20N 127036278 IC50 = 10.4 nM T56418 CQ9ZK4 127036284 IC50 = 16.4 nM T56418 CD4S5H 127036285 IC50 = 33 nM T56418 CWL9B0 127036286 IC50 = 9.5 nM T56418 C79URZ 127036287 IC50 = 40.3 nM T56418 C4INY9 127036288 IC50 = 11.2 nM T56418 C9MA2B 127036306 IC50 = 24 nM T56418 C4DT3E 127036344 IC50 = 1.7 nM T56418 C6QP8B 127036345 IC50 = 3.1 nM T56418 C1F9JZ 127036346 IC50 = 1.3 nM T56418 C09PRY 127036545 IC50 = 6.9 nM T56418 C6ZJR3 127036546 IC50 = 4.7 nM T56418 CUY1N9 127036698 IC50 = 32 nM T56418 C85AYL 127036893 IC50 = 11.8 nM T56418 CE61KB 127036900 IC50 = 21 nM T56418 CRG6Q3 127036901 IC50 = 38 nM T56418 CTN2Z5 127036902 IC50 = 381 nM T56418 CMI4B2 127036903 IC50 = 182 nM T56418 C0LG6K 127037082 IC50 = 53 nM T56418 CE4JU9 127037083 IC50 = 0.9 nM T56418 CZD87E 127037084 IC50 = 2 nM T56418 C9L3RE 127037085 IC50 = 7.1 nM T56418 C42NYM 127037086 IC50 = 4.6 nM T56418 C7C4RW 127037087 IC50 > 10000 nM T56418 C0OH9U 127037088 IC50 > 10000 nM T56418 C2HX8A 127037089 IC50 > 10000 nM T56418 CHG9Y4 127037090 IC50 > 10000 nM T56418 CY6CW4 127037091 IC50 > 10000 nM T56418 C8HMV5 127037291 IC50 > 10000 nM T56418 CVR06J 127042254 IC50 = 21 nM T56418 C38IPD 127045378 IC50 = 855 nM T56418 C09DVA 127045515 IC50 = 6203 nM T56418 CHK16Q 127045929 IC50 > 1000 nM T56418 CY3J0C 127047591 IC50 > 1000 nM T56418 CSEJ41 127048207 IC50 = 19 nM T56418 CDK3C6 127049147 IC50 = 1.86 nM T56418 C2MF9I 127049148 IC50 = 0.8 nM T56418 CV1E5D 127049149 IC50 = 4.77 nM T56418 C07TZN 127049440 IC50 = 0.75 nM T56418 C2FE1A 127049463 IC50 = 1.59 nM T56418 C7ODG2 127049464 IC50 = 0.99 nM T56418 C7A4OJ 127049465 IC50 = 0.59 nM T56418 CCP29E 127051596 IC50 = 291 nM T56418 C4WKQ5 127052926 IC50 = 59 nM T56418 CHQJ02 127052979 IC50 = 9.9 nM T56418 C9CVB0 129048532 IC50 = 12 nM T56418 CO1ST8 129065476 IC50 = 3.7 nM T56418 CXN46D 129148000 IC50 = 4.3 nM T56418 C8ZM1T 129281909 IC50 = 0.92 nM T56418 C97GOL 129896918 IC50 = 1.7 nM T56418 CUO0C5 132156633 IC50 > 10000 nM T56418 C4Q5LF 132471857 IC50 > 30000 nM T56418 C53OJM 132607333 IC50 = 2840.72 nM T56418 CMI3Q0 132819888 IC50 > 3333 nM T56418 CERS64 132937256 IC50 > 30000 nM T56418 C1WO9J 134132421 IC50 = 1.5 nM T56418 CTC53J 134134039 IC50 = 2.4 nM T56418 CPJG85 134135151 IC50 = 6.2 nM T56418 C9FZ3A 134136788 IC50 = 4.8 nM T56418 CG92RQ 134137314 IC50 = 73 nM T56418 C1U2MV 134137679 IC50 = 5.5 nM T56418 CHL7B1 134140023 IC50 = 67 nM T56418 C6M9DN 134140179 IC50 = 2.3 nM T56418 CPZU61 134140696 IC50 = 1.4 nM T56418 CW04KZ 134141466 IC50 = 6.1 nM T56418 C8KC5F 134142230 IC50 = 5.5 nM T56418 C9R3TS 134142441 IC50 = 7 nM T56418 CAL5D8 134145302 IC50 = 6.3 nM T56418 CQU86Z 134146557 IC50 = 7 nM T56418 CN35SO 134146628 IC50 = 1.5 nM T56418 CDCJ80 134148182 IC50 = 80 nM T56418 CFG60Q 134148895 IC50 = 9 nM T56418 CKOA84 134149727 IC50 = 17.1 nM T56418 C9Z1VM 134153244 IC50 = 30 nM T56418 C7H8GQ 134157229 IC50 = 9 nM T56418 CK5VG4 134219752 IC50 = 0.33 nM T56418 COL83G 134449962 IC50 = 36 nM T56418 CM56YZ 134449964 IC50 = 200 nM T56418 CYSD82 134449966 IC50 = 3.4 nM T56418 C50MOY 134449967 IC50 = 1.7 nM T56418 C8NHS5 134449968 IC50 = 6.1 nM T56418 CA1J8M 134449969 IC50 = 1.5 nM T56418 CKH86B 134449970 IC50 = 0.4 nM T56418 CMY2F8 134449972 IC50 = 1.5 nM T56418 CIDG30 134449973 IC50 = 2.1 nM T56418 CMH0E6 134449974 IC50 = 1.9 nM T56418 C53DWQ 134449975 IC50 = 1.4 nM T56418 C9G1LX 134449976 IC50 = 4 nM T56418 C4O6RT 134449977 IC50 = 2.2 nM T56418 CW1NP9 134449978 IC50 = 2.8 nM T56418 C5TO1D 134449980 IC50 = 1.9 nM T56418 C73XZL 134449984 IC50 = 2.1 nM T56418 C2PH8S 134449985 IC50 = 2.8 nM T56418 CV9CF2 134449987 IC50 = 1.7 nM T56418 CZ8W6R 134612705 IC50 = 3 nM T56418 CYL5V1 134694986 IC50 > 30000 nM T56418 C13ZRU 134817449 IC50 = 3.3 nM T56418 CM1XS0 135324340 IC50 = 11 nM T56418 CE8UF0 135483649 IC50 <= 99 nM T56418 CJI0G1 135520135 IC50 > 10000 nM T56418 CTJ48K 135524085 IC50 = 4100 nM T56418 CUT1W7 135524168 IC50 > 10000 nM T56418 CI47VJ 135566923 IC50 = 70 nM T56418 C0RXD7 135581817 IC50 = 239.49 nM T56418 CKW4C6 135873822 IC50 = 11 nM T56418 C8Y6ED 135957524 IC50 = 2400 nM T56418 C03MFU 135991097 IC50 <= 99 nM T56418 CHA4N2 136013680 IC50 > 10 nM T56418 C27WLC 136042304 IC50 = 392 nM T56418 C5YS8O 136042305 IC50 = 259 nM T56418 CPH0M8 136042306 IC50 = 7 nM T56418 CH64ID 136175114 IC50 > 10000 nM T56418 C1YUD0 136219394 IC50 > 10 nM T56418 CIU8W3 136254389 IC50 > 10 nM T56418 CSGM03 137210056 IC50 > 10000 nM T56418 CE75QD 137321162 IC50 > 10000 nM T56418 C31BFH 137347775 IC50 = 85 nM T56418 C7FVC0 137347776 IC50 = 17 nM T56418 CP4W5Q 137631562 IC50 = 2680 nM T56418 C25ERN 137631967 IC50 = 93.9 nM T56418 CZ8KV7 137632325 IC50 = 926 nM T56418 C39SCN 137632955 IC50 = 5.2 nM T56418 CI1E8V 137634241 IC50 > 10000 nM T56418 CPU3W0 137634339 IC50 = 8810 nM T56418 CMN0V1 137634592 IC50 = 190 nM T56418 CWO49T 137634681 IC50 = 58.8 nM T56418 CH7Z2E 137636265 IC50 = 21 nM T56418 C06JRX 137637094 IC50 = 101.1 nM T56418 C5C0ZR 137638616 IC50 = 118 nM T56418 C2ZXS7 137640634 IC50 = 310 nM T56418 CKOU26 137640983 IC50 = 41.5 nM T56418 C1G0VS 137641084 IC50 = 58 nM T56418 CIRS96 137642294 IC50 = 2860 nM T56418 CF4B3T 137642817 IC50 = 242 nM T56418 C3TIU9 137642961 IC50 = 4230 nM T56418 CA26QI 137644095 IC50 = 50.9 nM T56418 C09FUH 137644619 IC50 = 28.4 nM T56418 CF4R0S 137646760 IC50 = 26.3 nM T56418 C3L8VS 137647055 IC50 = 2710 nM T56418 CA01ZD 137647753 IC50 = 219 nM T56418 CE2WN1 137648666 IC50 = 5.3 nM T56418 CXS7O9 137649003 IC50 = 28400 nM T56418 C6AXN5 137649302 IC50 = 129 nM T56418 C1DK0P 137651391 IC50 = 155.5 nM T56418 CQ65AB 137652232 IC50 = 2700 nM T56418 C3Z4RJ 137652893 IC50 = 4740 nM T56418 C28AUH 137653585 IC50 = 93.5 nM T56418 C5F7TG 137654160 IC50 = 29 nM T56418 CDP3F4 137654891 IC50 = 377 nM T56418 CJC62Q 137655585 IC50 = 1.9 nM T56418 CL46TX 137656745 IC50 = 1180 nM T56418 C06XUG 137657541 IC50 = 547 nM T56418 C39KYU 137657831 IC50 = 30.7 nM T56418 CV5H3Z 137657932 IC50 = 231.1 nM T56418 CXC2L0 137658137 IC50 = 7130 nM T56418 C0B7RX 137658642 IC50 > 10000 nM T56418 CXH8P1 137660490 IC50 = 1483 nM T56418 CH12BE 138105933 IC50 = 20 nM T56418 C4Q9BD 138105934 IC50 = 2.5 nM T56418 C8A4ZC 138105936 IC50 = 2 nM T56418 CS8DI4 138108740 IC50 = 10 nM T56418 CWF2B5 138108958 IC50 = 10 nM T56418 CT1D9K 138454747 IC50 = 2100 nM T56418 C8WE0V 138454785 IC50 = 2.9 nM T56418 CT4A9I 138454797 IC50 = 18.72 nM T56418 CSRI06 138547901 IC50 > 1000 nM T56418 CUXO19 138617501 IC50 > 1000 nM T56418 COG63R 141482475 IC50 = 4700 nM T56418 CKN4Z9 141482476 IC50 = 7000 nM T56418 C1QZK2 141482477 IC50 = 9700 nM T56418 CX2TB0 141482479 IC50 = 3500 nM T56418 CFH6E9 141482480 IC50 > 10000 nM T56418 CWQ92I 141482481 IC50 = 9200 nM T56418 C16ZIH 141482484 IC50 = 6700 nM T56418 CPH01I 141482485 IC50 > 10000 nM T56418 C15RML 141482486 IC50 > 10000 nM T56418 CNR57A 141482487 IC50 = 1800 nM T56418 C5GEQ3 141482489 IC50 = 6700 nM T56418 C0FG1K 141482490 IC50 > 10000 nM T56418 C0UIW1 141482492 IC50 = 4500 nM T56418 CH9I3U 141482493 IC50 = 9600 nM T56418 C2DF4X 141482494 IC50 = 8700 nM T56418 CFE08V 141482495 IC50 = 7600 nM T56418 CJ61MC 141482496 IC50 > 10000 nM T56418 C34QYJ 141482498 IC50 = 8700 nM T56418 CC21GM 141482499 IC50 = 8000 nM T56418 C25PAE 141482501 IC50 > 10000 nM T56418 CQF23C 141482502 IC50 = 6800 nM T56418 CSK43T 141482503 IC50 = 4700 nM T56418 C0IBX2 141482504 IC50 = 2800 nM T56418 CSD1Z6 141488410 IC50 = 800 nM T56418 CVA4W1 141488417 IC50 = 2480 nM T56418 C34CKN 141523354 IC50 = 199.7 nM T56418 C6FH9Y 141727060 IC50 = 1.58 nM T56418 CD89PT 141727063 IC50 = 394.19 nM T56418 C84OXD 141727064 IC50 = 53.08 nM T56418 CPF28B 141727065 IC50 = 194.38 nM T56418 CB0AH8 141727069 IC50 = 253.18 nM T56418 CS1IQ9 141727073 IC50 > 2000 nM T56418 CT59SL 141727074 IC50 = 218.45 nM T56418 CLH67J 141727076 IC50 = 53.95 nM T56418 C0S1AY 141727077 IC50 = 83.15 nM T56418 CV7T9K 141727078 IC50 > 2000 nM T56418 CK7M8D 141727082 IC50 > 2000 nM T56418 CGHY63 141727083 IC50 = 94.05 nM T56418 C51RSN 141727084 IC50 = 648.59 nM T56418 CYP4D2 141727085 IC50 = 567.92 nM T56418 C19AUD 141727086 IC50 > 2000 nM T56418 COQR21 141727087 IC50 = 103.47 nM T56418 C2BY3V 141727090 IC50 = 27.05 nM T56418 CZ0YI7 141759648 IC50 = 1046 nM T56418 C29XUO 145945978 IC50 > 1000 nM T56418 C1AL7N 145949714 IC50 = 3100 nM T56418 CJ2SY5 145949745 IC50 = 7.8 nM T56418 CD3CH5 145949867 IC50 = 1.5 nM T56418 CGY21Q 145950006 IC50 = 10.5 nM T56418 CDZK73 145950618 IC50 = 8900 nM T56418 C6HC2M 145950676 IC50 > 10000 nM T56418 CBT87I 145950891 IC50 = 5900 nM T56418 CP5E1D 145951195 IC50 = 0.7 nM T56418 CQ2I5Y 145951801 IC50 = 6100 nM T56418 CM3CX8 145952650 IC50 = 4.3 nM T56418 C8V4MP 145952681 IC50 = 3 nM T56418 CVB73T 145952789 IC50 = 1.3 nM T56418 CMB03S 145953021 IC50 = 2.2 nM T56418 COA5Y3 145953378 IC50 = 2.3 nM T56418 C43OWV 145953418 IC50 = 6 nM T56418 C8LMR5 145953442 IC50 = 8100 nM T56418 CNE6Q7 145953506 IC50 = 83.2 nM T56418 C59WAN 145954203 IC50 = 3.3 nM T56418 CU9J0X 145954267 IC50 = 958 nM T56418 C89RPH 145954372 IC50 = 3.9 nM T56418 CA10CB 145954622 IC50 = 2300 nM T56418 CSA1N0 145955188 IC50 > 1000 nM T56418 CM3IY9 145955264 IC50 = 0.7 nM T56418 CV9M0Z 145955839 IC50 > 10000 nM T56418 C6A3QR 145956008 IC50 = 130 nM T56418 CROY34 145956057 IC50 = 24.2 nM T56418 C9CBZ7 145956245 IC50 = 6.9 nM T56418 C4C3FQ 145956510 IC50 = 0.8 nM T56418 C14ICP 145956607 IC50 = 6.2 nM T56418 CG5IT7 145956784 IC50 = 53.7 nM T56418 CXS07V 145956971 IC50 = 262 nM T56418 C20VAD 145957128 IC50 = 10.3 nM T56418 C2V8DA 145957160 IC50 = 4 nM T56418 C2O1TV 145957224 IC50 = 8600 nM T56418 C0O3PM 145958131 IC50 = 9500 nM T56418 C20XFU 145958474 IC50 = 2.6 nM T56418 C42ZQH 145958534 IC50 = 3.4 nM T56418 CXWH23 145958592 IC50 = 3 nM T56418 C79TLJ 145958973 IC50 = 48 nM T56418 C3TLJ8 145959766 IC50 = 8600 nM T56418 CR26HS 145959950 IC50 = 22.9 nM T56418 CQE9M5 145966810 IC50 = 190 nM T56418 CWJ12M 145969155 IC50 = 50 nM T56418 CGSA67 145971928 IC50 = 4.1 nM T56418 CDVM26 145971994 IC50 = 108 nM T56418 C2XDZ7 145972715 IC50 > 1000 nM T56418 CRP31S 145972920 IC50 = 4.2 nM T56418 CI6C4A 145973385 IC50 = 3600 nM T56418 CB4M6H 145973631 IC50 = 1 nM T56418 CS79NA 145974057 IC50 = 1.4 nM T56418 C74TYP 145975351 IC50 = 186.2 nM T56418 C4X8LC 145979928 IC50 = 2000 nM T56418 CNFJ75 145980559 IC50 = 4200 nM T56418 CJC1Z4 145980715 EC50 = 19630 nM T56418 CAE5G0 145987157 IC50 = 2200 nM T56418 C1J5IX 145990848 IC50 = 3900 nM T56418 C5KB0A 145991472 IC50 = 1600 nM T56418 CD30FP 145992021 Ki < 0.2 nM T56418 CGA41L 146014467 IC50 = 41.3 nM T56418 C60JPV 155166360 IC50 = 695 nM T56418 CL41OU 155183985 IC50 = 123 nM T56418 CPY92M 155510533 IC50 = 63 nM T56418 CV8SQ4 155510804 IC50 = 3.2 nM T56418 CB5X7K 155511395 IC50 = 270 nM T56418 CPZW51 155511600 IC50 = 520 nM T56418 C4PT8S 155511865 Ki < 0.02 nM T56418 C9VFI8 155512995 IC50 = 43 nM T56418 C2MD1Q 155513187 IC50 > 10000 nM T56418 CX4L3U 155516368 IC50 = 9.6 nM T56418 CCB4K6 155516809 IC50 = 338.51 nM T56418 C59EKB 155517980 IC50 = 757 nM T56418 CR68FM 155519610 IC50 = 0.87 nM T56418 CBY13X 155519739 IC50 = 17 nM T56418 CPS34K 155519748 IC50 = 210 nM T56418 C18ORE 155519760 IC50 = 14 nM T56418 CNU28S 155519814 IC50 = 3.7 nM T56418 CSP87Q 155519831 IC50 = 425.33 nM T56418 COQ7U0 155520571 IC50 = 17 nM T56418 C4L6HU 155521645 IC50 = 36.98 nM T56418 CLJ6B2 155522472 IC50 = 290 nM T56418 CGZ1N0 155523499 IC50 = 21 nM T56418 CZ56CF 155523941 IC50 = 350 nM T56418 CSRV18 155524183 IC50 = 2150 nM T56418 C4GR6U 155524577 IC50 = 558 nM T56418 CZ21UI 155525009 IC50 = 13.76 nM T56418 CQ0D4K 155525053 IC50 = 290 nM T56418 CLS4H2 155525411 IC50 = 440 nM T56418 CE5U8Z 155526528 IC50 = 560 nM T56418 CEF2G1 155526776 IC50 = 680 nM T56418 C9AG1S 155526843 IC50 = 1.9 nM T56418 CVQR59 155528115 IC50 = 1.2 nM T56418 C1QP6F 155528377 IC50 = 0.6 nM T56418 C7AS1F 155528651 IC50 = 47.4 nM T56418 CHI54P 155529236 IC50 = 11.5 nM T56418 C6VQ0W 155530641 IC50 = 2.7 nM T56418 CX7I1V 155531079 IC50 = 4.2 nM T56418 CVBK76 155531967 IC50 = 5.1 nM T56418 C3THR9 155532270 IC50 = 0.86 nM T56418 C8HDO1 155532442 IC50 = 38 nM T56418 CGVZ73 155532854 IC50 = 2.7 nM T56418 C1S6XO 155533569 IC50 = 490 nM T56418 C9JU0I 155534094 IC50 > 10000 nM T56418 CX91EL 155534287 IC50 = 413 nM T56418 CM0U3I 155534552 IC50 = 0.73 nM T56418 CX3AU5 155534611 IC50 = 492 nM T56418 CEQJ52 155534874 IC50 = 2.9 nM T56418 C78MZC 155536330 IC50 = 18 nM T56418 C3LC9I 155536820 IC50 = 5138 nM T56418 CRV8K0 155538035 IC50 = 4260 nM T56418 CL48RU 155538479 IC50 = 2 nM T56418 CH6Z8W 155538581 IC50 = 6.2 nM T56418 CLA3E7 155539013 IC50 > 2000 nM T56418 CCQ76W 155539390 IC50 = 661 nM T56418 CC3IQ7 155540048 IC50 = 103 nM T56418 CLD3F7 155540396 IC50 = 1.8 nM T56418 C80DML 155541340 IC50 = 3210 nM T56418 CI95ZY 155541415 IC50 = 336.38 nM T56418 CL6A7R 155541437 IC50 = 4340 nM T56418 C08QBJ 155541660 IC50 = 220 nM T56418 CT02GE 155541767 IC50 = 3.7 nM T56418 C0F5BN 155542940 IC50 = 0.27 nM T56418 C81WLX 155544983 IC50 = 1000 nM T56418 C46MQV 155546345 IC50 = 91 nM T56418 C7SF2C 155547229 IC50 > 10000 nM T56418 CBGI59 155547977 IC50 = 3.3 nM T56418 C60YKA 155548301 IC50 = 4.7 nM T56418 CW0YD8 155548579 IC50 = 43 nM T56418 CV20GX 155549214 IC50 = 250.94 nM T56418 CW19MB 155549248 IC50 = 0.64 nM T56418 C31NSY 155549763 IC50 = 129.9 nM T56418 CV7S6N 155550199 IC50 = 31 nM T56418 CE8LF0 155550275 IC50 = 370 nM T56418 C9J1MU 155550347 IC50 = 15 nM T56418 CZ4J2P 155552610 IC50 = 2.5 nM T56418 C0FH6Y 155554614 IC50 = 150 nM T56418 C31LPE 155555281 IC50 = 3400 nM T56418 CS4RB8 155557858 IC50 = 22 nM T56418 C1OI5K 155559863 IC50 = 0.91 nM T56418 CM3JG6 155561359 IC50 = 41 nM T56418 C1ZX4J 155563060 IC50 = 0.95 nM T56418 C7J9BO 155563111 IC50 = 14 nM T56418 C2ZI7W 155563158 IC50 = 42 nM T56418 CJN3Q9 155564067 IC50 = 2010 nM T56418 C6DAE5 155566754 IC50 = 21 nM T56418 CE79PT 155566881 IC50 = 39.64 nM T56418 C4QL2W 155567149 IC50 = 37 nM T56418 C4O8RS 155567235 IC50 = 370 nM T56418 CCP90I 155567914 IC50 = 0.6 nM T56418 D00ATA 5908088 IC50 > 50000 nM T56418 D02NZE 46871638 IC50 = 10 nM T56418 D03BQI 3794 IC50 = 2400 nM T56418 D03DZO 11715767 IC50 > 10000 nM T56418 D04CUA 44256277 IC50 = 340 nM T56418 D05MHL 44605611 Ki = 17 nM T56418 D06HVH 54613583 IC50 > 10000 nM T56418 D06PJW 25182616 IC50 = 0.5 nM T56418 D07OSK 6419834 IC50 = 5400 nM T56418 D08HFG 24809764 IC50 > 10000 nM T56418 D08TVU 46871653 IC50 = 150 nM T56418 D09HVH 135566652 IC50 > 10 nM T56418 D09PTP 57325421 IC50 = 1.9 nM T56418 D0CE3R 5312137 IC50 = 18000 nM T56418 D0E7VO 59627005 IC50 = 34.1 nM T56418 D0G4CS 25229528 IC50 = 14 nM T56418 D0H0LP 46906624 IC50 = 11 nM T56418 D0K5UF 72710568 Ki < 0.1 nM T56418 D0L4WN 31420 IC50 > 40000 nM T56418 D0O7LU 56599293 Ki = 0.75 nM T56418 D0R2WK 16038120 IC50 = 1.6 nM T56418 D0T8NU 16757525 IC50 > 4000 nM T56418 D0US9O 45275255 IC50 = 50 nM T56418 D0Y1UL 10561847 IC50 > 50000 nM T45074 CJWH47 127169 Ki = 24000 nM T45074 CODW17 192450 Ki = 8300000 nM T45074 CJC30Y 5071774 Ki = 4000000 nM T45074 CGV62F 10397086 Ki = 2600000 nM T45074 CZ6JA1 10442807 Ki = 25000000 nM T45074 CAFZ67 11819317 Ki = 1900000 nM T45074 CVP1W9 14545622 Ki = 7500000 nM T45074 C8I3OR 14545623 Ki = 20300000 nM T45074 C4Q9DV 44339325 Ki = 4100000 nM T45074 CG7F9J 44339646 Ki = 9200000 nM T92803 D05SBO 46220502 Ki < 10 nM T92803 D05ADP 160355 IC50 = 3000 nM T92803 D09JEJ 24748573 IC50 = 6.8 nM T92803 D0E3TC 44259 IC50 = 4.93 nM T92803 D0U2BH 65064 IC50 = 330 nM T92803 D00OWF 5280953 IC50 = 8.81 nM T92803 D02GEJ 5326976 IC50 = 400 nM T92803 D05BVP 3232621 IC50 = 27 nM T92803 D06MBI 1893668 IC50 = 12 nM T92803 D08DIJ 71529610 IC50 = 0.22 nM T92803 D09CDR 77105816 IC50 = 25 nM T92803 D09UNF 12248889 IC50 = 5500 nM T92803 D0CC7E 77105818 IC50 = 18 nM T92803 D0DT5I 71529599 IC50 = 0.98 nM T92803 D0GV3X 12248893 IC50 = 50 nM T92803 D0JQ0Z 46916176 IC50 = 17 nM T92803 D0NS6I 10037501 IC50 = 600 nM T92803 D0PJ1W 71529622 IC50 = 0.94 nM T92803 D0PO8N 117881270 IC50 = 104 nM T92803 D0Q3VZ 135398522 IC50 = 21 nM T92803 D0RG1T 44136031 IC50 = 240 nM T92803 D0WX0K 71680628 IC50 = 40 nM T92803 C1B9ZO 68094 IC50 = 90 nM T92803 CVMO57 95875 IC50 > 10000 nM T92803 CARD64 188439 IC50 = 66.7 nM T92803 CQU2B6 295893 IC50 > 10000 nM T92803 C34KZT 295897 IC50 > 10000 nM T92803 C12LUK 395921 IC50 = 11000 nM T92803 CVJC65 398318 IC50 > 10000 nM T92803 CFBU18 400433 IC50 = 588 nM T92803 C04FPT 486623 IC50 = 400 nM T92803 C7XM8E 621030 IC50 > 10000 nM T92803 CM3Y6Q 675788 IC50 = 6390 nM T92803 CS1YW9 705248 IC50 > 50000 nM T92803 CO3G5K 726514 IC50 = 2500 nM T92803 C1TFZ2 748299 IC50 > 50000 nM T92803 C3D1HC 762415 IC50 = 1810 nM T92803 C6GM9O 839804 IC50 = 2500 nM T92803 CKA4J5 851061 IC50 > 10000 nM T92803 C4YBX3 1003979 IC50 = 24740 nM T92803 CS6A9Q 1013797 IC50 = 19470 nM T92803 C8IQF6 1021429 IC50 = 20000 nM T92803 CS5L4Q 1104467 IC50 = 2500 nM T92803 CFA92X 1237489 IC50 = 1100 nM T92803 CD1A9T 1241605 IC50 = 250 nM T92803 C5QGK3 1270516 IC50 > 50000 nM T92803 CC7I1X 1350361 IC50 > 50000 nM T92803 CAV19R 2360773 IC50 > 10000 nM T92803 CM2Z4H 2807500 IC50 = 1510 nM T92803 CU80LI 3233012 IC50 = 98 nM T92803 CHCZ84 3233454 IC50 = 26000 nM T92803 C6NMC8 3233824 IC50 = 16420 nM T92803 CT8RJ2 3234850 IC50 = 1262 nM T92803 CW4C3P 3235048 IC50 > 10000 nM T92803 CSJ39A 3235398 IC50 = 5697 nM T92803 CP08XF 5179806 IC50 = 23710 nM T92803 CLM7V5 5371900 IC50 = 6400 nM T92803 CZU0A4 5479542 IC50 = 2200 nM T92803 CZ0NU2 5481591 IC50 = 35 nM T92803 CO6KI2 5930298 IC50 = 600 nM T92803 C1BNP3 9864573 IC50 = 16000 nM T92803 CG12HW 9881447 IC50 = 81 nM T92803 CJO47T 9948405 IC50 > 10000 nM T92803 CV8I5X 9999342 IC50 > 10000 nM T92803 CDCS35 10198544 IC50 = 8.8 nM T92803 C5TQ7X 10247543 IC50 > 10000 nM T92803 CU4Q9P 10268893 IC50 = 2100 nM T92803 C2WQ8M 10473563 IC50 > 10000 nM T92803 C81HMZ 11242728 IC50 > 10000 nM T92803 CBOP58 11293798 Ki > 10000 nM T92803 C26BZX 11362471 Ki > 10000 nM T92803 CWXB93 11397177 Ki > 10000 nM T92803 CTG83F 11539329 Ki > 6900 nM T92803 CACS26 11561968 Ki > 2000 nM T92803 CMIL86 11590363 Ki > 6900 nM T92803 C9T6SC 11640926 Ki > 6900 nM T92803 CP04JC 11666231 IC50 = 20 nM T92803 CU0E8O 11690457 Ki = 1000 nM T92803 CPI54D 11953235 IC50 = 14 nM T92803 CJ0NW4 12235681 IC50 = 200 nM T92803 CU5X3N 12248887 IC50 > 10000 nM T92803 CIDQ65 12248890 IC50 > 10000 nM T92803 CVG1Y9 12248891 IC50 > 10000 nM T92803 C2BD3Q 12248892 IC50 > 10000 nM T92803 CR3BS0 12248905 IC50 = 370 nM T92803 CN82LO 12448344 IC50 = 600 nM T92803 CD34SM 12456154 IC50 = 26000 nM T92803 CHJ01P 13303387 IC50 > 10000 nM T92803 C5YF0D 13303393 IC50 > 10000 nM T92803 CX27EP 13975510 IC50 = 1200 nM T92803 CFPW41 16007116 Ki > 6900 nM T92803 C5VPH9 16129448 IC50 = 2940 nM T92803 C3OP0J 16751208 IC50 = 406 nM T92803 CV7L6K 17942760 IC50 < 10000 nM T92803 CMW42V 19079253 IC50 = 1300 nM T92803 C48UIA 21413325 IC50 = 163 nM T92803 CG3VB6 23646578 IC50 = 110 nM T92803 CG6D4M 23647319 IC50 > 10000 nM T92803 CY8Z7X 23647330 IC50 > 10000 nM T92803 C4XD8H 23647348 IC50 > 10000 nM T92803 C7YG1N 24759534 IC50 < 10 nM T92803 CHLV09 24844836 IC50 = 971 nM T92803 CS81TH 24861908 IC50 > 100000 nM T92803 CLF9B0 25023078 IC50 = 4100 nM T92803 CW2YQ0 25141335 IC50 = 620 nM T92803 CS93BJ 25195482 IC50 = 2800 nM T92803 CX9M4Z 25211051 IC50 = 900 nM T92803 C8OK2N 27281959 IC50 = 3300 nM T92803 C71ZQL 29961826 IC50 > 50000 nM T92803 C8ICN3 44138082 IC50 = 600 nM T92803 CT0F8L 44142047 IC50 = 9012 nM T92803 C39AYP 44142048 IC50 > 10000 nM T92803 C18WIG 44142049 IC50 > 10000 nM T92803 CKZ91F 44142050 IC50 > 10000 nM T92803 C37NJT 44142051 IC50 = 4517 nM T92803 CI7K2Y 44142052 IC50 = 180 nM T92803 C3E4GY 44159452 IC50 = 2024 nM T92803 C2CY8P 44178895 IC50 = 4 nM T92803 CWH16X 44223933 IC50 = 3480 nM T92803 CGLQ20 44223952 IC50 = 206 nM T92803 CR6VH2 44223953 IC50 = 35 nM T92803 C2IBW0 44223954 IC50 = 541 nM T92803 CS3Q2Y 44223955 IC50 = 30 nM T92803 C5M1UN 44223957 IC50 = 120 nM T92803 C6E5PK 44223962 IC50 > 10000 nM T92803 CK8G1T 44223965 IC50 = 74 nM T92803 CJ8KD4 44223966 IC50 = 93 nM T92803 CCW0V4 44223967 IC50 = 155 nM T92803 CF78WD 44223968 IC50 = 1158 nM T92803 CNE30X 44223970 IC50 = 14 nM T92803 CYR45S 44223971 IC50 = 51 nM T92803 CLZ62P 44223973 IC50 = 31 nM T92803 CIXB09 44223974 IC50 = 57 nM T92803 C2OBX8 44223977 IC50 = 126 nM T92803 C62UWH 44456889 IC50 = 15000 nM T92803 C7OG2H 44591833 IC50 > 50000 nM T92803 CL2RP0 44591834 IC50 > 50000 nM T92803 CB3J0R 44591835 IC50 > 50000 nM T92803 CTU81O 44591836 IC50 = 1200 nM T92803 C1PR9H 44591837 IC50 > 50000 nM T92803 C02CVS 44591986 IC50 = 30000 nM T92803 C8SPN5 44592292 IC50 > 50000 nM T92803 CES0H7 44592293 IC50 > 50000 nM T92803 CO87DU 44592326 IC50 > 50000 nM T92803 CL87VC 44592327 IC50 = 20000 nM T92803 CP8L4V 44592328 IC50 > 50000 nM T92803 CUK90P 44592329 IC50 > 50000 nM T92803 C4FRI5 44592356 IC50 > 50000 nM T92803 CZ0PJ9 44592357 IC50 = 20000 nM T92803 CUO04L 44592358 IC50 > 50000 nM T92803 CBK5D9 44592359 IC50 = 15000 nM T92803 C07LQS 44592360 IC50 > 50000 nM T92803 C57JBM 44592426 IC50 = 5000 nM T92803 CWNG38 44592427 IC50 = 40000 nM T92803 CFL56G 44592495 IC50 = 600 nM T92803 CTRB87 44592496 IC50 > 50000 nM T92803 C34UTQ 44592497 IC50 > 50000 nM T92803 C4YAM7 44592498 IC50 > 50000 nM T92803 C8HTU7 44592499 IC50 > 50000 nM T92803 C1Z8UB 44592500 IC50 > 50000 nM T92803 CF9Z8L 44627215 IC50 > 10000 nM T92803 C87PSC 44820580 IC50 = 16400 nM T92803 C8O9RB 44820583 IC50 = 41200 nM T92803 CT69UN 44820586 IC50 = 26000 nM T92803 C7TLU8 44820588 IC50 = 32800 nM T92803 C7MRW5 44820589 IC50 = 46300 nM T92803 C6DG3M 44820595 IC50 = 29200 nM T92803 CI2J6V 44820597 IC50 = 20700 nM T92803 CW09EB 44820599 IC50 = 65400 nM T92803 CIWF96 44820602 IC50 = 41200 nM T92803 C3JBN1 44968184 IC50 = 260 nM T92803 CYW79D 44968186 IC50 = 38 nM T92803 CAY7V6 44968191 IC50 > 10000 nM T92803 C1RBX2 44968193 IC50 > 10000 nM T92803 C5OYK3 44968199 IC50 = 1437 nM T92803 COQ3X5 44968200 IC50 = 3152 nM T92803 CBS71N 44968204 IC50 > 10000 nM T92803 C2SI9M 44968206 IC50 = 164 nM T92803 CWY31S 44968208 IC50 > 10000 nM T92803 C2T0EM 44968221 IC50 = 3629 nM T92803 C8NA2J 44968224 IC50 = 1136 nM T92803 CR8DC5 44968225 IC50 = 922 nM T92803 CV19YK 44968230 IC50 = 557 nM T92803 CD4ZN1 44968231 IC50 > 10000 nM T92803 CQ0ZI7 45141513 IC50 = 13000 nM T92803 C3CF5U 45269374 IC50 > 10000 nM T92803 CEZL29 45269382 IC50 > 10000 nM T92803 CRE63M 45270204 IC50 > 10000 nM T92803 C0CT9X 45270205 IC50 > 10000 nM T92803 CSNR41 45271037 IC50 > 10000 nM T92803 C4UXH9 45271897 IC50 > 10000 nM T92803 C30UFN 45271898 IC50 > 10000 nM T92803 CG2DH1 45271903 IC50 > 10000 nM T92803 CIM9W4 45271904 IC50 > 10000 nM T92803 CJQU89 45273696 IC50 > 10000 nM T92803 C76HWN 46172958 IC50 = 6500 nM T92803 C6M9XJ 46172959 IC50 = 26000 nM T92803 CQUI12 46172960 IC50 = 26000 nM T92803 CT03XY 46172961 IC50 = 23200 nM T92803 CB0LE4 46172963 IC50 = 14600 nM T92803 CR74SM 46172965 IC50 = 29200 nM T92803 C16QFN 46172966 IC50 = 4654 nM T92803 C7J0IV 46172968 IC50 = 260 nM T92803 CE0W7X 46172970 IC50 = 26000 nM T92803 CB32ET 46172972 IC50 = 6361 nM T92803 CK1TI4 46172975 IC50 = 32800 nM T92803 C2AO9E 46172977 IC50 = 26000 nM T92803 CO90KZ 46172978 IC50 = 23200 nM T92803 CIHP23 46172979 IC50 = 29200 nM T92803 CN26HW 46172980 IC50 = 203 nM T92803 CJZ20M 46172982 IC50 = 20700 nM T92803 CLJZ24 46172983 IC50 = 32800 nM T92803 CGH05O 46172984 IC50 = 558 nM T92803 CN58VR 46172985 IC50 = 13000 nM T92803 CA40QS 46172989 IC50 = 29200 nM T92803 C65WIO 46172990 IC50 = 14600 nM T92803 CNJ2X9 46172991 IC50 = 26000 nM T92803 CY3HW5 46224684 IC50 = 440 nM T92803 C4X1BO 46316704 IC50 = 300 nM T92803 CLS29B 46872626 IC50 > 10000 nM T92803 CYBR24 46882056 IC50 = 410 nM T92803 C2O8RZ 46886323 IC50 > 1000 nM T92803 C0L5FV 46908045 IC50 > 10000 nM T92803 CQDV01 46908046 IC50 > 10000 nM T92803 C4DSY8 46908047 IC50 > 10000 nM T92803 CQ5HK0 46908048 IC50 > 10000 nM T92803 CM2Q8G 46908049 IC50 > 10000 nM T92803 CBI05Q 46908050 IC50 = 2400 nM T92803 C7A9BZ 46908051 IC50 > 10000 nM T92803 CTAB23 46909408 IC50 = 3400 nM T92803 CN0D2H 46909409 IC50 = 9000 nM T92803 CUO83H 46909508 IC50 = 4000 nM T92803 C3YE6Q 46909509 IC50 = 3500 nM T92803 C0DL3M 46909510 IC50 > 10000 nM T92803 CM70YK 46909511 IC50 > 10000 nM T92803 C5DW6Y 46909512 IC50 > 10000 nM T92803 CYB1V4 46909513 IC50 > 10000 nM T92803 C5K4TA 46909514 IC50 > 10000 nM T92803 CRLZ94 46912952 IC50 = 890 nM T92803 C1VA0B 46912953 IC50 = 710 nM T92803 C1PG7E 46912955 IC50 = 1100 nM T92803 C15EJK 46916169 IC50 > 10000 nM T92803 CHG8C4 46916170 IC50 = 70 nM T92803 CI56BA 46916172 IC50 = 26 nM T92803 CSFT47 46916173 IC50 = 4657 nM T92803 C93DCO 46916174 IC50 > 10000 nM T92803 CZ5DJ4 46916177 IC50 = 84 nM T92803 CXK37B 46916178 IC50 = 93 nM T92803 CL1GW0 46916179 IC50 = 76 nM T92803 CZ6DK4 46916182 IC50 = 135 nM T92803 C8BQ1W 46926509 IC50 = 26020 nM T92803 CR93YO 46926510 IC50 = 9230 nM T92803 C0FN2W 46926512 IC50 = 13040 nM T92803 CCUG10 46926515 IC50 = 107 nM T92803 C9NC6W 46926516 IC50 = 70 nM T92803 CZ1D2A 46926518 IC50 = 7 nM T92803 C7S6HT 46926519 IC50 = 18 nM T92803 CG1K5A 46926520 IC50 = 3454 nM T92803 CVF48X 46926521 IC50 = 25 nM T92803 C4ULH5 46926522 IC50 = 11 nM T92803 CPE98Z 46926523 IC50 = 26 nM T92803 C6WLX1 46926524 IC50 = 26020 nM T92803 CIU3B7 46926525 IC50 = 3280 nM T92803 C61LUI 46926526 IC50 = 273 nM T92803 C0IVD1 46926527 IC50 = 79 nM T92803 CE4SU5 47298428 IC50 = 100 nM T92803 CAYI59 49795862 IC50 = 1640 nM T92803 C1UQN4 49795863 IC50 = 2352 nM T92803 CU8OC0 49795864 IC50 = 1434 nM T92803 C7T5HW 49795865 IC50 = 61 nM T92803 C6N8EY 49795866 IC50 = 330 nM T92803 C7XS1Z 49795867 IC50 = 349 nM T92803 CR3LJ9 49795868 IC50 = 210 nM T92803 CLG75N 49831238 IC50 = 6300 nM T92803 C7LU5S 49838747 Ki = 1680 nM T92803 C6VQ7Y 49853605 IC50 > 10000 nM T92803 C20IFM 49854737 IC50 = 3300 nM T92803 CXI39D 49854741 IC50 = 1800 nM T92803 C4D3JF 49854742 IC50 = 6000 nM T92803 C5W3DH 49854744 IC50 = 1600 nM T92803 CAW0P1 49854960 IC50 > 10000 nM T92803 C9I4LQ 49855059 IC50 = 5500 nM T92803 C5EWG8 49855158 IC50 = 21 nM T92803 CD2K4R 50908681 Ki > 1000000 nM T92803 CVK96A 51351159 Ki = 252 nM T92803 CEQN27 52936621 Ki > 1000 nM T92803 C7AT0L 53316832 IC50 = 10000 nM T92803 C16VWZ 53318151 IC50 = 16000 nM T92803 CBH27E 53361525 IC50 = 79 nM T92803 CNA12Z 54575582 IC50 = 39 nM T92803 C65OUB 54575585 IC50 = 152 nM T92803 CS6N8Z 54581884 IC50 = 594 nM T92803 CO9QV2 54582429 IC50 = 21000 nM T92803 CYM84U 54766585 IC50 > 10000 nM T92803 CM31DA 54766737 IC50 = 21000 nM T92803 CH5OR4 54766892 IC50 = 43000 nM T92803 C3UC1Q 56929347 IC50 = 134 nM T92803 CDK93W 56946894 IC50 = 40 nM T92803 CZ1AP7 56956644 IC50 = 2300 nM T92803 C7ZD8T 57403741 IC50 = 88130 nM T92803 C3MFV7 57414126 IC50 = 5.9 nM T92803 CR3I5F 57418686 IC50 = 1400 nM T92803 CPK49W 57523834 IC50 = 780 nM T92803 CWB05Y 57523919 IC50 = 22 nM T92803 CW1CM5 57523921 IC50 = 41 nM T92803 C7K9YV 57523922 IC50 = 30 nM T92803 CB5MW8 57524010 IC50 = 305 nM T92803 C8N9SO 57524101 IC50 = 342 nM T92803 C45GPV 57524102 IC50 = 8 nM T92803 C6Z9FB 57524195 IC50 = 9 nM T92803 C91BAE 57524196 IC50 = 107 nM T92803 CPK6C8 57524269 IC50 = 12 nM T92803 C2XEQ5 57524335 IC50 = 47 nM T92803 CK2DM8 57524410 IC50 = 156 nM T92803 CJ91XM 57524491 IC50 = 6 nM T92803 C4O0QZ 57524820 IC50 = 116 nM T92803 CTID23 57524821 IC50 = 97 nM T92803 C3KRE2 57524829 IC50 = 1610 nM T92803 CQM73T 57524896 IC50 = 180 nM T92803 CFH12N 57524901 IC50 = 9 nM T92803 C4WGF1 57524903 IC50 = 1030 nM T92803 CVTB94 58047131 IC50 = 900 nM T92803 CPW8T1 58221748 IC50 = 1300 nM T92803 CF6K1Y 58857683 IC50 = 9400 nM T92803 C3ZPO8 58880668 IC50 > 10000 nM T92803 C56MAG 59379853 IC50 = 7800 nM T92803 C4S6HC 59581274 IC50 = 1 nM T92803 CXJ63M 59603829 IC50 = 11 nM T92803 CQEU96 59603842 IC50 = 3.2 nM T92803 C1MR8Q 60097495 IC50 > 1000 nM T92803 C8CP1H 60155996 Ki = 158 nM T92803 C6NF3R 60161879 IC50 = 59 nM T92803 CIS84M 60162923 IC50 = 320 nM T92803 C37NKO 67129970 IC50 = 4860 nM T92803 CK80LJ 67130050 IC50 > 10000 nM T92803 C3MF9D 67134733 IC50 = 80000 nM T92803 C1SB2C 67134967 IC50 = 93000 nM T92803 CHN3F1 67135258 IC50 >= 10000 nM T92803 C6AG1I 67135489 IC50 = 25000 nM T92803 C7X1CW 67135729 IC50 = 4500 nM T92803 C9HZR2 67135774 IC50 = 2200 nM T92803 CV63UL 67240318 IC50 > 10000 nM T92803 CO4FB2 67283393 IC50 > 10000 nM T92803 CUQ4Z2 67283468 IC50 > 10000 nM T92803 CA13ZR 67283600 IC50 > 10000 nM T92803 C9LDM1 67283615 IC50 > 10000 nM T92803 C94IJP 67283623 IC50 > 10000 nM T92803 CLX0Q2 67283821 IC50 > 10000 nM T92803 CN79BL 67283829 IC50 > 10000 nM T92803 CQY7C6 67283926 IC50 > 10000 nM T92803 CY0CW9 67284258 IC50 = 50000 nM T92803 C59ZIA 67284569 IC50 > 10000 nM T92803 C4S7VO 67284820 IC50 > 10000 nM T92803 C56LDY 67471491 IC50 > 10000 nM T92803 C7YNV0 67471492 IC50 > 10000 nM T92803 CT5BE6 67471493 IC50 > 10000 nM T92803 CHQ1Z0 68034378 Ki = 2015 nM T92803 CKY3W6 68108530 IC50 = 797 nM T92803 CYW71X 68108891 IC50 = 9 nM T92803 COPZ25 68108932 IC50 = 13 nM T92803 C9VMR0 68109014 IC50 = 37 nM T92803 C6PE0H 68109248 IC50 = 52 nM T92803 C0COB2 68109381 IC50 = 301 nM T92803 CB8SP0 68109626 IC50 = 15 nM T92803 C7GRV2 68755406 IC50 > 10000 nM T92803 C5DGR9 69036886 IC50 = 10000 nM T92803 C0T1JU 69069650 IC50 = 3300 nM T92803 COL1Q7 70370469 IC50 = 1229 nM T92803 CQA3B0 70370554 IC50 = 5 nM T92803 C3WK5U 70684923 IC50 = 790 nM T92803 CN8T9F 70695463 IC50 = 1600 nM T92803 CCM6X2 71272330 IC50 = 5.1 nM T92803 CFU0O9 71277772 IC50 = 194.4 nM T92803 C5JHE3 71277785 IC50 = 26.2 nM T92803 C82UAF 71450223 IC50 > 10000 nM T92803 CMSG37 71450224 IC50 = 7600 nM T92803 C51WVQ 71450225 IC50 > 10000 nM T92803 CJNF34 71452050 IC50 > 10000 nM T92803 C2ZNM4 71452051 IC50 > 10000 nM T92803 CDA2V4 71452052 IC50 > 10000 nM T92803 C3G2FA 71453864 IC50 = 1800 nM T92803 CAR9O2 71453865 IC50 > 10000 nM T92803 C53XMV 71455595 IC50 = 8100 nM T92803 CKT60L 71455860 Ki > 6800 nM T92803 CQSW87 71457381 IC50 > 10000 nM T92803 C6ATV1 71457382 IC50 = 5600 nM T92803 CBV9D5 71517518 IC50 > 10000 nM T92803 C5E4PU 71517519 IC50 > 10000 nM T92803 CV7D6Y 71517520 IC50 = 5300 nM T92803 C1X7IP 71517683 IC50 = 9000 nM T92803 C4GEZ7 71517684 IC50 = 3400 nM T92803 CHJ6Y4 71517685 IC50 = 2000 nM T92803 CLYA16 71517686 IC50 = 1200 nM T92803 C6F2YJ 71517687 IC50 = 1000 nM T92803 C3POF4 71517688 IC50 = 1100 nM T92803 C1LA5R 71517855 IC50 = 400 nM T92803 CQ4BW8 71517856 IC50 = 400 nM T92803 CRG30M 71517858 IC50 = 800 nM T92803 CNXZ69 71517859 IC50 = 780 nM T92803 CDPM84 71517860 IC50 = 900 nM T92803 C1E2WR 71517861 IC50 > 10000 nM T92803 CQL58Z 71518030 IC50 = 2000 nM T92803 CBO84W 71518031 IC50 > 10000 nM T92803 C1LZH0 71518032 IC50 = 7000 nM T92803 C1CLS7 71518033 IC50 = 3200 nM T92803 C6GSA0 71518034 IC50 = 2800 nM T92803 CJH3Q6 71518035 IC50 = 1000 nM T92803 CTP65Y 71518036 IC50 = 1100 nM T92803 C24VAR 71518204 IC50 = 280 nM T92803 C2DG7M 71518205 IC50 = 270 nM T92803 C1XMB9 71518206 IC50 = 300 nM T92803 CTXS51 71518207 IC50 = 490 nM T92803 CZ81WY 71518373 IC50 = 450 nM T92803 CDU08C 71518374 IC50 = 300 nM T92803 CE1FT3 71518375 IC50 = 280 nM T92803 CVI5T9 71518530 IC50 = 480 nM T92803 C0DCR9 71518533 IC50 = 480 nM T92803 COB76S 71529590 IC50 = 436.1 nM T92803 CY30GN 71529591 IC50 = 9.53 nM T92803 C4OP6Q 71529598 IC50 = 1.81 nM T92803 CA8T4S 71529600 IC50 = 6.06 nM T92803 CW9CI7 71529601 IC50 = 42.7 nM T92803 C70TAN 71529603 IC50 = 3.89 nM T92803 C4IS7N 71529612 IC50 = 39.03 nM T92803 C9UTB3 71529613 IC50 = 13.64 nM T92803 C5OPK8 71529614 IC50 = 35.64 nM T92803 C1RP0Y 71529624 IC50 = 18.26 nM T92803 CQ4GS7 71529626 IC50 = 6.02 nM T92803 CG5EZ4 71529627 IC50 = 33.93 nM T92803 CIDV86 71529733 IC50 = 431.2 nM T92803 CW63BV 71529753 IC50 = 13.08 nM T92803 CPQU78 71529756 IC50 = 1.65 nM T92803 C3VAQ2 71608036 IC50 = 3.6 nM T92803 CT5VG6 71716749 IC50 = 1000 nM T92803 CC1IL9 71717349 IC50 = 4000 nM T92803 CZ13FJ 71717350 IC50 = 300 nM T92803 C7KY6G 71717351 IC50 = 1900 nM T92803 C09KIW 71717352 IC50 = 1200 nM T92803 C3S4DL 71717942 IC50 = 16000 nM T92803 CT18BN 71717943 IC50 = 5800 nM T92803 C4KJ6M 71717944 IC50 = 3900 nM T92803 CY05XE 71719167 IC50 = 2500 nM T92803 CLOH34 71719168 IC50 = 3800 nM T92803 CZ2XE3 71719776 IC50 = 2100 nM T92803 CQ2B7A 71720387 IC50 = 3000 nM T92803 C8JD6S 71720388 IC50 = 500 nM T92803 C7ZW9K 71720389 IC50 = 400 nM T92803 C1QO3R 71745026 IC50 > 10000 nM T92803 CNOX90 72700319 IC50 = 110 nM T92803 CBY80T 72716071 IC50 = 30000 nM T92803 CAQ87R 72724765 IC50 > 10000 nM T92803 CB1EX4 72724904 IC50 = 6520 nM T92803 C36SAZ 72725030 IC50 = 4010 nM T92803 CYLK14 73333219 IC50 = 440 nM T92803 C0T6IK 73345875 IC50 = 0.99 nM T92803 CD6G8Z 73347380 IC50 = 0.36 nM T92803 C2AG9F 73425095 IC50 = 443 nM T92803 C4BV9L 73426232 IC50 > 1000 nM T92803 CV6XS5 73707532 Ki = 575 nM T92803 CO15QH 76309392 IC50 = 2000 nM T92803 CY32ES 76313100 IC50 = 2000 nM T92803 CVD5U4 76314850 IC50 = 500 nM T92803 C1U0SR 76314852 IC50 = 830 nM T92803 C61JOY 76314853 IC50 = 1800 nM T92803 CY23ZG 76316620 IC50 = 500 nM T92803 C1FNZ6 76316622 IC50 = 2300 nM T92803 CS82OQ 76320341 IC50 = 650 nM T92803 CN0JZ3 76320342 IC50 = 800 nM T92803 C2WL9U 76320343 IC50 = 1100 nM T92803 CMKG91 76323973 IC50 = 2100 nM T92803 CIB1A6 76323974 IC50 = 510 nM T92803 CBE1L4 76324679 IC50 = 17000 nM T92803 C3UM1R 76325751 IC50 = 3100 nM T92803 C0KY3T 76327523 IC50 = 4700 nM T92803 C8KN6T 76327524 IC50 = 3000 nM T92803 CBW95G 76327525 IC50 = 3200 nM T92803 C1T5HL 76327526 IC50 = 1100 nM T92803 C3YH9Q 76331196 IC50 = 710 nM T92803 C9RX0H 76331198 IC50 = 1000 nM T92803 CAQW90 76331199 IC50 = 3000 nM T92803 CZD34Y 76331200 IC50 = 1200 nM T92803 C63MTJ 76334790 IC50 = 7000 nM T92803 CVZ58T 76334791 IC50 = 1200 nM T92803 C21JAS 76853169 IC50 = 870 nM T92803 CW64MP 77105434 IC50 = 1200 nM T92803 CU04XY 77105624 IC50 = 180 nM T92803 C3NX4F 77105815 IC50 = 600 nM T92803 CEW7R1 77105817 IC50 = 2000 nM T92803 CIM47W 77105819 IC50 = 3300 nM T92803 CTIA65 77105820 IC50 = 970 nM T92803 CH79MO 77105821 IC50 = 670 nM T92803 CKB1P9 77106023 IC50 = 27 nM T92803 CTP6N7 77106024 IC50 = 4000 nM T92803 CXYW85 77106025 IC50 = 310 nM T92803 C2UDS0 77106026 IC50 = 850 nM T92803 C97SJD 77106027 IC50 = 600 nM T92803 CFQ10R 77106028 IC50 = 370 nM T92803 CO14DP 77106030 IC50 = 850 nM T92803 C5GM2W 77106233 IC50 > 10000 nM T92803 C9G3PA 77106234 IC50 = 5800 nM T92803 CPD27I 77106235 IC50 = 4300 nM T92803 CLOR37 77106236 IC50 = 200 nM T92803 C2GLD8 77106237 IC50 = 440 nM T92803 C8D3XO 86765295 IC50 = 5700 nM T92803 C0GYK1 86765296 IC50 = 75 nM T92803 COQ7N2 87338044 IC50 = 8700 nM T92803 CE28YU 87338241 IC50 >= 10000 nM T92803 CTG02V 87338507 IC50 > 10000 nM T92803 C9ND7G 87411868 IC50 > 10000 nM T92803 CT6AI0 87411870 IC50 > 10000 nM T92803 C9XMG6 87411871 IC50 > 10000 nM T92803 C4BKA6 89429109 IC50 = 7300 nM T92803 C2FOK4 89494280 IC50 = 650 nM T92803 C1HW4B 89735655 IC50 = 130 nM T92803 CB40PI 90306552 IC50 > 10000 nM T92803 CE5L8V 90388565 IC50 = 2400 nM T92803 CCAN79 90645088 IC50 > 10000 nM T92803 CE5M0Z 90645089 IC50 > 10000 nM T92803 CUY63S 90645193 IC50 > 10000 nM T92803 C26BSU 90666124 IC50 = 1300 nM T92803 CVQ1O6 90666126 IC50 = 700 nM T92803 C5AN9J 90666128 IC50 = 1800 nM T92803 CP76NE 90666130 IC50 > 10000 nM T92803 C85GHD 90666131 IC50 > 10000 nM T92803 CRP9I5 90666132 IC50 > 10000 nM T92803 CWE9I2 91664021 IC50 = 6 nM T92803 CW58AE 91664022 IC50 = 180 nM T92803 CB25UZ 91664023 IC50 = 120 nM T92803 CNC4Q0 91664024 IC50 = 181 nM T92803 C3KJ8R 98073446 IC50 = 55.2 nM T92803 CL64EZ 102287891 IC50 > 10000 nM T92803 C2NQ4S 102287892 IC50 > 10000 nM T92803 C5N1VZ 102581295 IC50 > 10000 nM T92803 C7XUO9 118450030 IC50 = 7957 nM T92803 C8G5IT 118714396 IC50 = 400 nM T92803 CB8G1T 118714397 IC50 = 3100 nM T92803 CEB3G4 118714398 IC50 = 15000 nM T92803 CTUZ03 118714399 IC50 = 3400 nM T92803 CRV8H7 118714400 IC50 = 3400 nM T92803 C7PAU6 118714401 IC50 = 9700 nM T92803 C6FQ8M 118714402 IC50 = 200 nM T92803 CXK5C3 118714403 IC50 = 11000 nM T92803 CJ89SC 118714404 IC50 = 2000 nM T92803 C1GU9B 118714405 IC50 = 1200 nM T92803 CF2IE6 118714406 IC50 = 6000 nM T92803 C2ZBH0 118714407 IC50 = 2000 nM T92803 CZ3G9V 118714408 IC50 = 42000 nM T92803 CK64OD 118714410 IC50 = 2900 nM T92803 CJF80M 118715634 IC50 > 10000 nM T92803 CLC5I4 118715635 IC50 > 10000 nM T92803 CDX07C 118715636 IC50 = 5100 nM T92803 CT6UF9 118715637 IC50 > 10000 nM T92803 CMG5I0 118715638 IC50 = 610 nM T92803 C4DQX9 118735337 IC50 = 19 nM T92803 CV01GL 118737103 IC50 = 530 nM T92803 C8GB4Q 122181008 IC50 = 2600 nM T92803 CBQ94Z 122181009 IC50 > 10000 nM T92803 CT8CP2 122181010 IC50 > 10000 nM T92803 CB6IZ0 122181011 IC50 > 10000 nM T92803 C65BOF 122181012 IC50 > 10000 nM T92803 CO83PN 122181013 IC50 = 31 nM T92803 C69ULZ 122181014 IC50 = 20 nM T92803 CN14DV 122181015 IC50 = 32 nM T92803 CIG8Y1 122181016 IC50 = 320 nM T92803 CRJS41 122181017 IC50 = 23 nM T92803 CVB03H 122181018 IC50 = 18 nM T92803 C6SJ3X 122181019 IC50 = 22 nM T92803 C8IM5O 122181020 IC50 = 2300 nM T92803 C7L5PG 122181021 IC50 = 2000 nM T92803 C58CJI 122181022 IC50 = 10000 nM T92803 CG2Z8B 122181023 IC50 = 39 nM T92803 CC2G8N 122181024 IC50 = 41 nM T92803 CM2DU7 122181025 IC50 = 56 nM T92803 C5YB3O 122181096 IC50 = 170 nM T92803 CV5BQ9 122181097 IC50 = 130 nM T92803 C5KB1C 122184057 IC50 = 100 nM T92803 C2XC3U 122187688 IC50 > 10000 nM T92803 C1WM3S 122187689 IC50 = 34000 nM T92803 C16YOP 122187742 IC50 > 10000 nM T92803 CC92DV 122187743 IC50 > 10000 nM T92803 CG13AW 122187744 IC50 > 10000 nM T92803 C5MPV3 122187745 IC50 = 7000 nM T92803 CI19TJ 122187746 IC50 > 10000 nM T92803 CJ9ZX6 122187747 IC50 > 10000 nM T92803 CLQ51W 122187748 IC50 > 10000 nM T92803 C8M3JO 122187749 IC50 = 6200 nM T92803 CL4Q8W 122187750 IC50 > 10000 nM T92803 CBK46E 122187751 IC50 > 10000 nM T92803 CY64GW 122187797 IC50 > 10000 nM T92803 CVBF01 127030212 IC50 = 170 nM T92803 CI93ZA 127030213 IC50 = 880 nM T92803 C8LQV4 127030516 IC50 = 1080 nM T92803 CS12RU 127031435 IC50 = 40 nM T92803 C0O9MC 127031570 IC50 > 10000 nM T92803 CZXP62 127031750 IC50 = 930 nM T92803 C3E5YO 127032014 IC50 = 130 nM T92803 C2ZD8S 127032024 IC50 = 700 nM T92803 CXWY73 127032324 IC50 = 960 nM T92803 C9H5VJ 127032841 IC50 = 7100 nM T92803 CZK6Y5 127032842 IC50 = 3000 nM T92803 CGUM96 127033730 IC50 = 3600 nM T92803 C5XR1J 127033735 IC50 > 10000 nM T92803 C8G6RH 127033736 IC50 > 10000 nM T92803 CZ6RJ5 127033737 IC50 > 10000 nM T92803 COEW54 127033738 IC50 > 10000 nM T92803 C1QX5Y 127034001 IC50 = 2800 nM T92803 C2P4ZJ 127034002 IC50 = 5100 nM T92803 CKWS32 127034003 IC50 > 10000 nM T92803 C2O9JK 127034004 IC50 > 10000 nM T92803 CX4OM5 127034021 IC50 > 10000 nM T92803 C2WJK8 127034519 IC50 = 4600 nM T92803 C1FZY7 127034520 IC50 = 4700 nM T92803 C2LWZ1 129318964 IC50 = 138 nM T92803 COW21D 129762063 IC50 = 54.8 nM T92803 C4W6AD 129897084 IC50 = 340 nM T92803 C3LR4A 134130122 IC50 = 5000 nM T92803 CAW7I8 134130909 IC50 > 10000 nM T92803 CW84QM 134131222 IC50 > 10000 nM T92803 C6B0RL 134131311 IC50 = 7300 nM T92803 CNJ15A 134132649 IC50 > 10000 nM T92803 C7D9WS 134132677 IC50 = 2600 nM T92803 C1UIL9 134135426 IC50 > 10000 nM T92803 C9EQC4 134136966 IC50 > 10000 nM T92803 C4AXE1 134140955 IC50 = 6000 nM T92803 CXA1S4 134142195 IC50 = 8900 nM T92803 CGC6D7 134143498 IC50 > 10000 nM T92803 CSHZ53 134145427 IC50 = 4700 nM T92803 C13TBI 134149173 IC50 > 10000 nM T92803 CP1BV6 134149357 IC50 = 4000 nM T92803 C3HO1K 134152098 IC50 = 3000 nM T92803 CZ65XP 134154248 IC50 > 10000 nM T92803 CE42VG 134156031 IC50 > 10000 nM T92803 C8WIV6 134157974 IC50 > 10000 nM T92803 C2AN7T 134611886 IC50 > 100000 nM T92803 CD57GW 134812697 Ki = 104 nM T92803 CNYW80 134812698 Ki > 2800 nM T92803 C07ODH 134812699 Ki = 383 nM T92803 CM8DK3 134813913 IC50 = 120 nM T92803 CGBZ13 134843302 IC50 > 10000 nM T92803 CR1E5Y 135335801 IC50 = 8 nM T92803 CGO0L8 135335871 IC50 = 7 nM T92803 CUG3X6 135335915 IC50 = 6 nM T92803 CJ7FM6 135335919 IC50 = 4 nM T92803 C09BEG 135486057 IC50 > 10000 nM T92803 CPCA46 135566559 IC50 = 7.6 nM T92803 CJBU04 135590713 IC50 = 10000 nM T92803 CBU0J4 135604653 IC50 > 100000 nM T92803 CG9R0V 135741827 IC50 > 10000 nM T92803 C12JNY 135909380 IC50 = 32 nM T92803 CM81HG 136044188 IC50 = 220 nM T92803 CT6N1O 136044189 IC50 > 10000 nM T92803 C9PTA8 136044190 IC50 = 1500 nM T92803 CM1EN4 136044191 IC50 > 10000 nM T92803 C5RI6D 136224254 IC50 > 10000 nM T92803 CT9VC6 136224366 IC50 > 10000 nM T92803 CF6B3S 136224367 IC50 > 10000 nM T92803 CH0Q2Z 136234577 IC50 = 50 nM T92803 CV6F4N 136234578 IC50 = 28 nM T92803 C2G3JY 136234579 IC50 = 8500 nM T92803 CC7Q8V 136238871 IC50 = 5000 nM T92803 C1JZ7D 136241623 IC50 = 27400 nM T92803 C1TGM4 136244455 IC50 = 8.63 nM T92803 C6S1GT 136245126 IC50 > 10000 nM T92803 CS6K0B 136245127 IC50 > 10000 nM T92803 CA5KP8 136245128 IC50 > 10000 nM T92803 CLF3B0 136259623 IC50 = 4.91 nM T92803 C8UQ7C 136264319 IC50 > 10000 nM T92803 CNE6I8 136264499 IC50 > 10000 nM T92803 CJC89A 136333957 IC50 = 59 nM T92803 CRB3M4 136609929 IC50 = 230 nM T92803 C0A9VE 136609930 IC50 = 470 nM T92803 CW5YL0 136609931 IC50 = 840 nM T92803 C3MK9W 136807986 IC50 > 10000 nM T92803 CCAZ26 137631656 IC50 = 110 nM T92803 CBJ2Q7 137631708 IC50 = 277 nM T92803 C3QAV9 137631819 IC50 = 1000 nM T92803 CQ15NR 137631839 IC50 = 7000 nM T92803 CK5WC1 137632241 IC50 = 790 nM T92803 CI43OC 137632412 IC50 = 204 nM T92803 CBPE50 137632517 IC50 = 2142 nM T92803 CV2B1M 137632742 IC50 = 2939 nM T92803 C7RAH4 137632779 IC50 < 10000 nM T92803 CG8Y0U 137633419 IC50 = 11000 nM T92803 C7E1FL 137633791 IC50 = 245 nM T92803 CH4PN9 137633814 IC50 = 31 nM T92803 C3BZK6 137633859 IC50 = 404 nM T92803 CVL41R 137633869 IC50 = 12 nM T92803 CS9TU2 137633985 IC50 = 930 nM T92803 CI1E8V 137634241 IC50 > 10000 nM T92803 C83UKG 137634382 IC50 = 340 nM T92803 CI73CB 137634638 IC50 = 3356 nM T92803 CNT7S3 137634818 IC50 = 5100 nM T92803 CCP7X5 137635304 IC50 = 2800 nM T92803 C1AK8X 137635556 IC50 = 2800 nM T92803 CV7OF5 137635713 IC50 = 1800 nM T92803 CQ2I7Y 137635832 IC50 > 10000 nM T92803 C5QWE1 137635926 IC50 = 39 nM T92803 C8GQD5 137636872 IC50 = 6.5 nM T92803 CW9K4H 137636941 IC50 = 8 nM T92803 C97FAW 137637167 IC50 = 1756 nM T92803 CM7N8S 137637724 IC50 = 1303 nM T92803 CKZF46 137638065 IC50 = 4400 nM T92803 CRV1E4 137638175 IC50 > 1000 nM T92803 CCX37E 137638472 IC50 = 93 nM T92803 CPO87L 137638509 IC50 = 57 nM T92803 C7CP2N 137638906 IC50 < 10000 nM T92803 C1UI5N 137638944 IC50 = 1400 nM T92803 C4XEI1 137639320 IC50 = 138 nM T92803 CH4RP3 137639514 IC50 = 510 nM T92803 CX3MQ1 137639546 IC50 = 120 nM T92803 C89JWP 137639612 IC50 > 10000 nM T92803 CH3S8N 137640038 IC50 = 33 nM T92803 C84RSO 137640193 IC50 = 257 nM T92803 CXM4G7 137640811 IC50 = 390 nM T92803 CF83TG 137640934 IC50 = 110 nM T92803 CB86PD 137641220 IC50 = 46 nM T92803 C3CE9O 137641621 IC50 = 194 nM T92803 CRSQ71 137641785 IC50 = 86 nM T92803 CI17FX 137641801 IC50 = 62 nM T92803 CGCF41 137642917 IC50 = 1337 nM T92803 CWVE69 137643514 IC50 = 580 nM T92803 CPO60W 137643573 IC50 > 10000 nM T92803 C7XN6Z 137643596 IC50 = 94 nM T92803 CYA1F7 137643721 IC50 = 120 nM T92803 C2AG3W 137643887 IC50 = 14000 nM T92803 C4DS3I 137643955 IC50 = 2500 nM T92803 C75MLQ 137643957 IC50 = 56 nM T92803 CWIP72 137644498 IC50 = 350 nM T92803 C74DEQ 137644716 IC50 = 242 nM T92803 CZ4U0W 137644802 IC50 = 220 nM T92803 CDA2N6 137644922 IC50 = 53 nM T92803 CPJ42V 137644974 IC50 > 10000 nM T92803 CWM1P5 137645266 IC50 = 1139 nM T92803 C0OTG4 137645459 IC50 = 75 nM T92803 C8VTQ9 137645650 IC50 = 3200 nM T92803 C7ZOV3 137645947 IC50 > 10000 nM T92803 CDE8O3 137646031 IC50 = 3360 nM T92803 CL5NX9 137646497 IC50 = 710 nM T92803 CJ5O2Q 137646673 IC50 = 3100 nM T92803 CK6S5T 137646758 IC50 > 1000 nM T92803 COU37W 137647335 IC50 = 50 nM T92803 C21IMP 137647416 IC50 < 10000 nM T92803 CMI2H3 137647526 IC50 = 169 nM T92803 COW27K 137647779 IC50 = 1 nM T92803 C7O2AW 137647969 IC50 > 10000 nM T92803 C7J9VR 137648478 IC50 > 10000 nM T92803 CCNA21 137648707 IC50 = 520 nM T92803 CNW13G 137648784 IC50 = 344 nM T92803 CGK5P2 137649037 IC50 = 212 nM T92803 CS69XL 137649171 IC50 = 500 nM T92803 C5OJH2 137649318 IC50 = 78 nM T92803 CM50YV 137649413 IC50 = 420 nM T92803 C9IO5F 137649821 IC50 = 6.6 nM T92803 CP9EN8 137650185 IC50 = 61 nM T92803 C9QNG8 137650421 IC50 = 9000 nM T92803 CW04TZ 137650486 IC50 = 89 nM T92803 CWG94C 137650926 IC50 = 2200 nM T92803 C8MKN0 137651314 IC50 = 470 nM T92803 CKL0P4 137651538 IC50 = 2100 nM T92803 CJ14XO 137651668 IC50 = 1500 nM T92803 CR0L9E 137651705 IC50 > 10000 nM T92803 CB1H3L 137651798 IC50 > 10000 nM T92803 CH6L2T 137652047 IC50 = 420 nM T92803 CI8TV2 137652861 IC50 = 351 nM T92803 C2B5CY 137652970 IC50 = 1600 nM T92803 C48DVU 137653000 IC50 = 190 nM T92803 CB6RP0 137653080 IC50 = 285 nM T92803 C01URE 137653446 IC50 = 1700 nM T92803 CDX83M 137654129 IC50 = 43 nM T92803 C47FBV 137654225 IC50 = 2100 nM T92803 CTBD05 137654245 IC50 = 1318 nM T92803 CX7V6P 137654671 IC50 > 1000 nM T92803 C1U5PD 137654853 IC50 = 10 nM T92803 CQC49I 137654914 IC50 = 2872 nM T92803 C8TDA4 137655242 IC50 = 109 nM T92803 C7D9PN 137655679 IC50 = 177 nM T92803 C7IU4J 137655848 IC50 = 79 nM T92803 CN1DW2 137655950 IC50 = 107 nM T92803 CYQ61R 137656593 IC50 = 1000 nM T92803 CQEJ60 137656868 IC50 = 63 nM T92803 C9M5WS 137657239 IC50 = 141 nM T92803 C3Y2CR 137657691 IC50 = 280 nM T92803 CN39CD 137657748 IC50 = 4335 nM T92803 C0SBY3 137657758 IC50 > 10000 nM T92803 CA10CX 137657812 IC50 = 127 nM T92803 C39SEV 137658150 IC50 = 1100 nM T92803 CX8YL9 137658187 IC50 = 75 nM T92803 CD73NA 137658280 IC50 = 283 nM T92803 CC34LO 137658348 IC50 = 8 nM T92803 CTO04D 137658447 IC50 < 10000 nM T92803 CX4M8T 137658722 IC50 > 1000 nM T92803 CA2PY1 137658970 IC50 = 470 nM T92803 CJ1TB2 137659239 IC50 = 7900 nM T92803 C3U2OB 137659350 IC50 = 870 nM T92803 CAF68S 137659391 IC50 > 10000 nM T92803 CFL9P1 137659439 IC50 < 10000 nM T92803 CXE25G 137659488 IC50 = 69 nM T92803 C0U2ZV 137659586 IC50 > 10000 nM T92803 C7QM6B 137659788 IC50 < 10000 nM T92803 CR98AD 137660581 IC50 > 10000 nM T92803 CD9W1H 137660657 IC50 = 2904 nM T92803 C7MI2G 137661183 IC50 = 4200 nM T92803 CIX41F 137661315 IC50 = 8900 nM T92803 CD0FV8 137661355 IC50 = 1300 nM T92803 C9HPG8 137661516 IC50 = 140 nM T92803 CT3F1E 139512365 IC50 = 49.5 nM T92803 C2KB4M 139520309 IC50 = 25 nM T92803 C1T0AO 139520310 IC50 = 13.9 nM T92803 C9BAN7 140682661 IC50 = 7.9 nM T92803 CHN0D8 145950829 IC50 = 858 nM T92803 CWY6T4 145950977 IC50 = 123 nM T92803 CM7Q1A 145952573 IC50 = 264 nM T92803 C2C1KB 145958797 IC50 = 159 nM T92803 CI0W7J 145958822 IC50 = 1500 nM T92803 CG1BN8 145971214 IC50 = 221 nM T92803 CENA85 145979136 IC50 = 18 nM T92803 C2B7VE 145979242 IC50 = 101 nM T92803 C2OF0R 145980649 IC50 = 14.9 nM T92803 C6ZQL2 145981774 IC50 = 29.7 nM T92803 C53HBS 145981791 IC50 = 4.6 nM T92803 CXD83F 145985653 IC50 = 63 nM T92803 CO1S8D 145986658 IC50 = 420000 nM T92803 CC8DY2 145987190 IC50 = 51.4 nM T92803 C1L3UE 145988000 IC50 = 106.7 nM T92803 CWUH96 145988043 IC50 = 90.5 nM T92803 CTWD68 145988875 IC50 = 14.3 nM T92803 CWP60I 145989404 IC50 = 42.6 nM T92803 C84YFW 145989761 IC50 = 130 nM T92803 COG96W 145990023 IC50 = 6 nM T92803 C17QCK 145990660 IC50 = 107 nM T92803 C0BW5M 145990753 IC50 = 23.5 nM T92803 C1MUA8 145991360 IC50 = 76 nM T92803 CPK48V 145991505 IC50 = 614.3 nM T92803 CZU8J6 145992124 IC50 = 3.2 nM T92803 C2CFU8 145992307 IC50 = 5 nM T92803 CK56CB 145993150 IC50 = 95 nM T92803 CI65VR 145993339 IC50 = 183.2 nM T92803 C39SMA 145993393 IC50 = 43 nM T92803 CQ48WH 145993525 IC50 = 57.8 nM T92803 C5YW8Q 145993622 IC50 = 2.1 nM T92803 CA0I5S 145993962 IC50 = 49 nM T92803 CN8GC1 145994089 IC50 = 37.3 nM T92803 CWE2R0 155513125 IC50 = 97 nM T92803 C2MD1Q 155513187 IC50 > 10000 nM T92803 CRB4Y7 155513451 IC50 = 215 nM T92803 CVZ0N8 155515881 IC50 = 19 nM T92803 CYV5T2 155525879 IC50 = 27 nM T92803 CTLN05 155538036 IC50 = 168 nM T92803 C68GMW 155538446 IC50 > 10000 nM T92803 CZ1OA4 155538975 IC50 = 112 nM T92803 C78ADU 155539435 IC50 = 56 nM T92803 CFMX59 155540359 IC50 = 168 nM T92803 CGZ86V 155542559 IC50 = 64 nM T92803 CF1PW9 155545528 IC50 = 1020 nM T92803 CGV45S 155545839 IC50 = 10 nM T92803 C3N9OK 155550070 IC50 = 950 nM T92803 CY6Q8S 155554337 IC50 > 10000 nM T92803 CHS3J0 155555099 IC50 = 13 nM T92803 CFUO14 155555367 IC50 = 98 nM T92803 C1NK2F 155559198 IC50 = 83.5 nM T92803 C75NXB 155559880 IC50 = 139 nM T92803 CO2I4P 155559898 IC50 = 2300 nM T92803 CUY6L4 155565201 IC50 = 74 nM T92803 D00AQR 71529770 IC50 = 1.13 nM T92803 D00ERW 44444843 Ki = 3401 nM T92803 D00HVA 11624601 Ki > 6900 nM T92803 D01MNK 25125014 IC50 = 2100 nM T92803 D06CXU 46926513 IC50 = 50 nM T92803 D07OAT 456214 IC50 = 300 nM T92803 D08NQM 5289247 IC50 = 30 nM T92803 D09ZNV 447682 IC50 = 8000 nM T92803 D0A1CM 5281855 IC50 > 40000 nM T92803 D0CP3M 5149739 IC50 = 2100 nM T92803 D0I1FJ 11393719 IC50 = 4900 nM T92803 D0L4WN 31420 IC50 = 3600 nM T92803 D0O1YH 1694 IC50 < 1000 nM T92803 D0Q3NG 11715520 Ki > 6900 nM T92803 D0S7IE 11658882 Ki > 6900 nM T92803 D0UI7U 46926514 IC50 = 2600 nM T92803 D0X9PI 71529752 IC50 = 0.16 nM T92803 D0Y5RO 4566 IC50 = 900 nM T24634 D01GYT 446987 IC50 = 100 nM T24634 D08UVZ 68423 IC50 = 7800 nM T24634 CS1KR4 72724 IC50 > 50000 nM T24634 CT2YS5 73174 IC50 > 50000 nM T24634 CKV26X 5849412 IC50 = 2800 nM T24634 C19ORL 11273626 IC50 = 9600 nM T24634 CTY4W5 11435907 IC50 = 27300 nM T24634 CY5D6A 44400303 IC50 > 50000 nM T24634 C6H1UC 44400324 IC50 = 9900 nM T24634 CC0W8S 44400490 IC50 = 20100 nM T24634 CQR0O7 44400556 IC50 > 50000 nM T24634 CF51RI 44400564 IC50 > 50000 nM T24634 COW7U2 44400587 IC50 > 50000 nM T24634 C7CE9D 44419231 IC50 > 50000 nM T24634 CC9MZ0 52948006 IC50 = 16700 nM T24634 CRXF52 54679840 IC50 = 1 ug.mL-1 T24634 CXKE26 54682555 IC50 > 25 ug.mL-1 T24634 C8UN1J 54712725 IC50 = 17 ug.mL-1 T24634 C39MDC 54728582 IC50 > 25 ug.mL-1 T24634 CHC41J 54728583 IC50 = 2 ug.mL-1 T24634 CXQ08D 54728584 IC50 = 3 ug.mL-1 T24634 CPU1Q7 54728585 IC50 > 25 ug.mL-1 T24634 C8OAV0 54728586 IC50 = 1 ug.mL-1 T24634 C3Q4ZU 54728587 IC50 > 25 ug.mL-1 T24634 CYF20S 54728588 IC50 = 14 ug.mL-1 T24634 C70FLC 54728589 IC50 > 25 ug.mL-1 T24634 C26FBM 54728590 IC50 = 5 ug.mL-1 T24634 C0SXV7 54728591 IC50 > 25 ug.mL-1 T24634 CK0BJ9 54728592 IC50 = 16 ug.mL-1 T24634 CWS12N 54728593 IC50 = 20 ug.mL-1 T24634 CONQ08 54728594 IC50 > 25 ug.mL-1 T24634 C1Q3YH 54728595 IC50 > 25 ug.mL-1 T24634 C69NOJ 54728596 IC50 = 4 ug.mL-1 T24634 C9CGU2 54728597 IC50 = 2 ug.mL-1 T24634 CGXT73 54728598 IC50 = 17 ug.mL-1 T24634 CA19RH 54728599 IC50 = 10 ug.mL-1 T24634 C2G9XV 54728600 IC50 = 1 ug.mL-1 T24634 C4LQ7K 54728603 IC50 > 25 ug.mL-1 T24634 CAWP39 54728605 IC50 > 25 ug.mL-1 T24634 COFR80 54728606 IC50 = 3 ug.mL-1 T24634 CW0L3M 54728607 IC50 > 25 ug.mL-1 T24634 C4U1RG 54728608 IC50 = 4 ug.mL-1 T24634 CR2S0C 108068 IC50 > 50000 nM T24634 D06HIW 5281461 IC50 = 32700 nM T24634 D07KNG 5281437 IC50 > 50000 nM T24634 D0S2TZ 119093 IC50 = 19500 nM T55610 D02PMO 60700 EC50 = 12 nM T55610 D06GKR 2973 EC50 = 17800 nM T55610 D06ZVO 11234794 IC50 = 20200 nM T55610 D00GOM 71453910 IC50 = 2150 nM T55610 D0K0PG 16124726 IC50 = 2440 nM T55610 D07HTX 148091 IC50 = 1 nM T55610 CN37HD 6842 IC50 = 1000 nM T55610 CYWS98 185848 IC50 > 50000 nM T55610 CQC5E6 362401 IC50 = 35200 nM T55610 CLUP70 991507 IC50 = 430 nM T55610 CW7K5I 1730746 IC50 = 2600 nM T55610 C2HX4K 2217157 EC50 = 20000 nM T55610 C2XN5M 2779853 IC50 = 43 nM T55610 CCVF41 2962284 EC50 = 7720 nM T55610 C60FMS 3236125 EC50 = 8850 nM T55610 CC21YG 3555371 IC50 = 3000 nM T55610 CL0CT4 3906683 IC50 = 5030 nM T55610 CF70TK 5124065 IC50 = 350 nM T55610 CKC6I5 5280462 IC50 = 15800 nM T55610 C4H5FJ 6404644 EC50 = 4480 nM T55610 CO53KT 6404645 EC50 = 7460 nM T55610 C84CTS 6413024 EC50 = 4620 nM T55610 C8PRK4 10030510 IC50 = 20 nM T55610 CEOI54 10084880 IC50 = 6100 nM T55610 CN1EO4 11267663 EC50 = 35000 nM T55610 C7HK0A 11305157 IC50 = 7500 nM T55610 CFQ42U 11525980 IC50 > 30000 nM T55610 CID2P7 11536421 IC50 > 30000 nM T55610 CAUL10 11559627 IC50 = 90 nM T55610 CF28TK 11565353 IC50 > 30000 nM T55610 CEG5W8 11608830 IC50 > 30000 nM T55610 CEO14D 11680638 IC50 = 810 nM T55610 CZK16N 14539883 IC50 = 0.14 nM T55610 CBA1K3 14539884 IC50 = 0.65 nM T55610 CNI19E 15479637 IC50 = 1030 nM T55610 C7QJO4 15479638 IC50 = 1260 nM T55610 C5U3GA 15944763 IC50 = 270 nM T55610 C0SG2C 16124727 IC50 = 3100 nM T55610 CI3QD6 20056162 IC50 = 140 nM T55610 C21ZEX 22970306 IC50 = 9160 nM T55610 CXPL52 24779732 IC50 = 600 nM T55610 CD7WK9 24779733 IC50 = 4100 nM T55610 C2ZF5A 24811989 IC50 = 1030 nM T55610 CBLW69 24811990 IC50 = 5000 nM T55610 CN3I8F 25154309 IC50 = 1800 nM T55610 CYN34U 25184847 IC50 > 30000 nM T55610 CT4A8I 25184848 IC50 > 30000 nM T55610 C4Q6TW 25184849 IC50 = 8000 nM T55610 C29PRB 25184907 IC50 > 30000 nM T55610 C2BHM3 25184908 IC50 > 30000 nM T55610 CZ5MI8 25184910 IC50 = 15000 nM T55610 CSW5G1 25184911 IC50 = 30000 nM T55610 C5UN2D 25184912 IC50 > 30000 nM T55610 CK8Y3G 25184913 IC50 = 8000 nM T55610 CO3TS9 25184970 IC50 = 1400 nM T55610 C3R1OG 25208124 IC50 = 0.65 nM T55610 CF15DX 25208125 IC50 = 5880 nM T55610 C4YNU8 34829688 EC50 = 16600 nM T55610 CJR6U2 42604718 IC50 = 6.76 nM T55610 C5TGC0 44224203 IC50 = 32500 nM T55610 CZX51L 44434920 IC50 = 820 nM T55610 C2QXA5 44434921 IC50 = 3400 nM T55610 C4AO7M 44434922 IC50 > 30000 nM T55610 C6B1IA 44443250 IC50 = 800 nM T55610 C6ABE2 44443251 IC50 > 30000 nM T55610 CZ43LE 44443253 IC50 = 3400 nM T55610 C2LKD9 44443254 IC50 = 900 nM T55610 CH5AO0 44443256 IC50 = 2500 nM T55610 CN43WG 44443257 IC50 > 30000 nM T55610 C7TX0Q 44443259 IC50 = 1300 nM T55610 C5W3AG 44443261 IC50 = 1900 nM T55610 CP2M6V 44443262 IC50 = 900 nM T55610 CWI4H7 44446962 IC50 = 214 nM T55610 CGJ60Y 44602318 EC50 = 3040 nM T55610 C05IBC 44602350 EC50 = 3080 nM T55610 C1MTJ6 44602351 EC50 = 2390 nM T55610 CDRW67 44602352 EC50 = 1190 nM T55610 C2D4RE 44631782 EC50 = 4270 nM T55610 C0T8HU 44631783 EC50 = 2460 nM T55610 C8JPW4 44631784 EC50 = 2480 nM T55610 C30XJG 44631785 EC50 = 10500 nM T55610 CK58PR 44631786 EC50 = 11600 nM T55610 CIUZ86 44631790 EC50 = 9080 nM T55610 C3OK9H 44631792 EC50 = 6270 nM T55610 CJQK09 45099939 EC50 = 3260 nM T55610 CZWR28 45099942 EC50 = 5410 nM T55610 C3BTG2 45099947 EC50 = 8690 nM T55610 C45RQB 45485201 IC50 = 4100 nM T55610 CM61JZ 45791805 IC50 = 7210 nM T55610 C7OA9C 46232839 IC50 = 3100 nM T55610 CI6YN2 46232840 IC50 = 4600 nM T55610 CM3JP5 46232841 IC50 = 90600 nM T55610 CX7J3D 46232842 IC50 = 91800 nM T55610 C6OQ5B 46232961 IC50 > 100000 nM T55610 CB1W5L 46232962 IC50 = 70400 nM T55610 C1QL8C 46232963 IC50 = 35300 nM T55610 C1EPZ8 46232964 IC50 > 100000 nM T55610 C3QTS6 46232965 IC50 > 100000 nM T55610 CDC63W 46233004 IC50 > 100000 nM T55610 C3FW6S 46233005 IC50 = 84800 nM T55610 C8EOL5 46233006 IC50 = 40300 nM T55610 CX04BM 46742338 EC50 = 1850 nM T55610 C6YO3P 46742340 EC50 = 1490 nM T55610 CPLI91 46742341 EC50 = 3670 nM T55610 CM82LV 46742342 EC50 = 3920 nM T55610 C5WG6X 46742343 EC50 = 2060 nM T55610 CVT8K6 46742344 EC50 = 1200 nM T55610 CX7TA6 46742345 EC50 = 600 nM T55610 CUB5A4 46742347 EC50 = 4350 nM T55610 C0OQ3E 46742349 EC50 = 3630 nM T55610 CCIB51 46742350 EC50 = 6450 nM T55610 CFRV57 46742351 EC50 = 9600 nM T55610 CMQ25T 46742353 EC50 = 1120 nM T55610 CKH6W5 46742354 EC50 = 500 nM T55610 CA38QS 46742355 EC50 = 7670 nM T55610 CD9IN2 46848332 IC50 = 690 nM T55610 CGV03O 47443232 IC50 = 55700 nM T55610 CW81OM 53248886 IC50 = 1 nM T55610 C4-MAY-02 53304209 IC50 > 30000 nM T55610 CPCN01 53304210 IC50 > 30000 nM T55610 C3CU6Z 53304211 IC50 > 30000 nM T55610 C5SPK4 53304212 IC50 = 2600 nM T55610 CS2E7L 53304213 IC50 = 7300 nM T55610 C7ECY9 53304214 IC50 = 12900 nM T55610 C8SQU9 53304383 IC50 = 5300 nM T55610 C13MTW 53304384 IC50 = 16800 nM T55610 C3TC6P 53304385 IC50 = 17200 nM T55610 CIM4R1 53304386 IC50 = 17500 nM T55610 CG98LW 53306268 IC50 = 10 nM T55610 CB6EU3 53306269 IC50 = 46 nM T55610 COQ7W5 53306270 IC50 = 4.2 nM T55610 CUZE47 53306271 IC50 = 54 nM T55610 C6NE5D 53306433 IC50 = 490 nM T55610 CR1FD6 53306434 IC50 = 580 nM T55610 C8ZGS2 53306435 IC50 = 7 nM T55610 CT5RX7 53306436 IC50 = 110 nM T55610 C7EO9I 53306437 IC50 = 54 nM T55610 CVB3C7 53306438 IC50 = 310 nM T55610 CZE43R 53306439 IC50 = 360 nM T55610 CMC5Q1 53306580 IC50 = 1100 nM T55610 CND4X6 53306581 IC50 > 30 nM T55610 C9ERA8 53306582 IC50 > 30000 nM T55610 CYS92X 53306583 IC50 = 26200 nM T55610 CM4QO9 53306584 IC50 > 30000 nM T55610 C6F9CU 53306585 IC50 > 30000 nM T55610 CA8OX7 53306586 IC50 > 30000 nM T55610 CJZT82 54580396 IC50 = 69900 nM T55610 CH83IB 54580397 IC50 > 100000 nM T55610 CL5ZQ3 54581400 IC50 = 51700 nM T55610 CZ0CY9 54581401 IC50 = 18700 nM T55610 C0XK3E 54581402 IC50 = 8620 nM T55610 C48BRQ 54583397 IC50 = 23000 nM T55610 CNX68C 54583398 IC50 = 41600 nM T55610 C5B7HI 54584345 IC50 = 22100 nM T55610 CTF9E7 54584346 IC50 = 15100 nM T55610 C5V0FB 54585313 IC50 = 32700 nM T55610 CP3BM7 54586264 IC50 = 17400 nM T55610 CKVM73 54586265 IC50 = 52100 nM T55610 C0LE7W 54587289 IC50 = 35500 nM T55610 CCK97R 54587290 IC50 > 100000 nM T55610 CX5WT3 54587291 IC50 = 39100 nM T55610 CW23ZV 54587292 IC50 = 29600 nM T55610 CFE5A9 56657947 IC50 = 470 nM T55610 CC1J0Q 56659540 IC50 > 30000 nM T55610 CWUK24 56661479 IC50 = 1200 nM T55610 C6CT9I 56664909 IC50 = 810 nM T55610 CCF30U 56666256 IC50 = 4200 nM T55610 C2DB0U 56666257 IC50 = 22900 nM T55610 CN8CW2 56666258 IC50 = 3500 nM T55610 CL18JY 56668337 IC50 = 160 nM T55610 C6BU1C 56669667 IC50 = 3300 nM T55610 C7J0BX 56671829 IC50 = 27600 nM T55610 CX6MQ9 56673175 IC50 = 4100 nM T55610 C7YXM4 56675402 IC50 = 27600 nM T55610 CRWY02 56679819 IC50 = 200 nM T55610 CMFZ90 56681867 IC50 = 1700 nM T55610 CTU87V 56681868 IC50 = 9400 nM T55610 CV6IY2 56681869 IC50 = 27500 nM T55610 CQ7O8T 56683148 IC50 = 6200 nM T55610 C2CUJ8 56683370 IC50 = 17600 nM T55610 CSIW76 56967243 IC50 = 740 nM T55610 C1DE4B 56967303 IC50 = 6030 nM T55610 CAW89I 56967304 IC50 = 1040 nM T55610 CY8H6V 56967305 IC50 = 4120 nM T55610 C20VHM 56967306 IC50 = 2170 nM T55610 C7DE6O 56967307 IC50 = 2380 nM T55610 CK5U8A 56967308 IC50 = 1180 nM T55610 CCJ26V 56967366 IC50 > 20000 nM T55610 C9F1JZ 56967367 IC50 > 20000 nM T55610 C74QFZ 56967368 IC50 = 820 nM T55610 CVO2S4 56967369 IC50 = 1840 nM T55610 C95IDN 56967370 IC50 = 1350 nM T55610 CM14OW 56967432 IC50 = 120 nM T55610 COV6R7 56967433 IC50 > 20000 nM T55610 C81UQV 56967434 IC50 > 20000 nM T55610 CT0UR7 56967435 IC50 = 1070 nM T55610 C2TO4C 56967436 IC50 = 1340 nM T55610 CM4GZ1 56967495 IC50 = 1850 nM T55610 C61BPZ 70291363 IC50 = 2870 nM T55610 COS48U 70701596 IC50 = 1400 nM T55610 C1YN7T 71453683 IC50 = 2540 nM T55610 C91EDL 71457190 IC50 > 20000 nM T55610 C75JWS 71457421 IC50 = 1360 nM T55610 CX6J2N 71459048 IC50 = 15750 nM T55610 CB7YS8 71462558 IC50 = 2620 nM T55610 CT0CP7 71488794 IC50 = 3 nM T55610 C39ZWP 71625259 IC50 = 14 nM T55610 C4QLE2 71716241 IC50 > 30000 nM T55610 C9KM4F 71717477 IC50 > 30000 nM T55610 CGIR31 71718067 IC50 = 270 nM T55610 CU54QR 71720505 IC50 = 3200 nM T55610 CMO1W9 71720506 IC50 = 34 nM T55610 C8LG0W 73293539 IC50 = 4300 nM T55610 C2R1QU 73349944 IC50 = 3800 nM T55610 C1QI8E 73443066 IC50 = 4700 nM T55610 CMQ73W 90488965 IC50 = 1900 nM T55610 CK1Y7S 101885530 EC50 = 2300 nM T55610 CHKZ09 118723281 IC50 > 30000 nM T55610 C6UIS1 118723282 IC50 > 30000 nM T55610 CGC5Z8 118723283 IC50 > 30000 nM T55610 C7M3PR 118723284 IC50 = 11400 nM T55610 CWUF31 118723285 IC50 > 30000 nM T55610 CM82UG 118723286 IC50 > 30000 nM T55610 CEF7L2 122179606 EC50 = 6700 nM T55610 CV5AM0 122179619 EC50 = 1400 nM T55610 CFS5I6 122179620 EC50 = 6700 nM T55610 CTJU67 122179621 EC50 = 15500 nM T55610 CMS62A 122179622 EC50 = 7800 nM T55610 CMC2B5 122179623 EC50 = 4100 nM T55610 CF64QK 122700533 IC50 = 12030 nM T55610 C8H6YS 122700551 IC50 = 940 nM T55610 CMK2L7 122700570 IC50 = 8450 nM T55610 CJ0NL2 122700638 IC50 = 360 nM T55610 CF0X9H 122700639 IC50 = 1330 nM T55610 CM0S7K 122700642 IC50 = 6350 nM T55610 CK9XQ2 122700667 IC50 = 100 nM T55610 C2SX7W 122700669 IC50 = 820 nM T55610 CG5IA1 122700672 IC50 = 880 nM T55610 CPRH14 122700678 IC50 = 1440 nM T55610 C80MDI 122700783 IC50 = 790 nM T55610 C3R8WD 122700873 IC50 = 3210 nM T55610 C3W4RE 122701004 IC50 = 1020 nM T55610 CB8K2A 122701008 IC50 = 1270 nM T55610 C06IAY 122701021 IC50 = 6210 nM T55610 C2UE7C 122701031 IC50 = 2880 nM T55610 CHTS12 127048856 IC50 = 29900 nM T55610 CAC7Z6 127048857 IC50 = 50000 nM T55610 C42YLJ 127052576 IC50 = 41700 nM T55610 CCS18G 132938257 IC50 = 12500 nM T55610 C9MW7D 135324866 IC50 = 1400 nM T55610 CF0D4J 135407624 IC50 = 8300 nM T55610 CAW0J5 135451013 IC50 = 730 nM T55610 CI3F5V 135876029 IC50 = 3 nM T55610 CUAR37 135909391 IC50 > 30000 nM T55610 C9VT0K 135909392 IC50 > 30000 nM T55610 CUEA47 135909406 IC50 > 30000 nM T55610 C4OK9P 135909407 IC50 = 5500 nM T55610 CJV8D0 135909408 IC50 > 30000 nM T55610 CN4JU5 135909409 IC50 = 5500 nM T55610 C1UEY7 135909410 IC50 = 800 nM T55610 C58WAG 135909413 IC50 = 6000 nM T55610 CFEN86 135909414 IC50 > 30000 nM T55610 CH7U5R 135909416 IC50 = 1500 nM T55610 C8JGA0 135909419 IC50 > 30000 nM T55610 CAO12C 135909420 IC50 = 4000 nM T55610 CW2H5S 135909421 IC50 > 30000 nM T55610 C57JFQ 136002677 IC50 = 2000 nM T55610 CY7S6E 136002678 IC50 > 30000 nM T55610 CA1ZS4 136721264 IC50 > 100000 nM T55610 C57YWQ 137287454 IC50 = 2400 nM T55610 CMJR40 137287455 IC50 = 2200 nM T55610 C0MJ7V 137633077 IC50 > 40000 nM T55610 CU2EI0 137633266 IC50 = 1120 nM T55610 CY57XU 137633414 IC50 = 29400 nM T55610 CUA0O2 137633479 IC50 = 1080 nM T55610 CF6QH3 137638733 IC50 = 45400 nM T55610 C8O4MI 137638756 IC50 = 27100 nM T55610 C5E4WV 137640233 IC50 = 25600 nM T55610 CY2B7I 137640646 IC50 = 870 nM T55610 C5SX0M 137640936 IC50 = 4520 nM T55610 CI3A9U 137641216 IC50 = 36300 nM T55610 CJQ2P0 137641683 IC50 = 34100 nM T55610 CODJ07 137643513 IC50 = 600 nM T55610 CD4P7F 137644657 IC50 = 36200 nM T55610 CL06XM 137645510 IC50 = 20800 nM T55610 C6NPL0 137645630 IC50 = 19900 nM T55610 CW68TH 137646187 IC50 = 15500 nM T55610 C42KBF 137647413 IC50 = 22600 nM T55610 CHK4R6 137648461 IC50 > 40000 nM T55610 CG4LJ9 137650328 IC50 = 19400 nM T55610 CIXM67 137653045 IC50 = 32700 nM T55610 CM2WX1 137653081 IC50 = 14880 nM T55610 CIPR91 137653603 IC50 > 20000 nM T55610 CJH40R 137658630 IC50 = 16500 nM T55610 CS35FI 137659032 IC50 = 3400 nM T55610 C5TX6S 137659436 IC50 = 24400 nM T55610 CS3U5X 137659554 IC50 = 45400 nM T55610 CW4R8O 137659784 IC50 = 36600 nM T55610 CDCM73 137660764 IC50 = 940 nM T55610 CQ1P0N 139600307 IC50 = 320 nM T55610 CGQ8U7 141467461 IC50 = 550 nM T55610 C71ZXB 141467463 IC50 = 620 nM T55610 CSQ6N2 142736726 IC50 > 15000 nM T55610 C32OGH 145964826 IC50 = 2820 nM T55610 CCJR12 145965591 IC50 = 3410 nM T55610 CV9H3T 145965757 IC50 = 2610 nM T55610 CT94UP 145966056 IC50 = 3150 nM T55610 CKWN80 145966486 IC50 = 1850 nM T55610 CT0RE4 145967305 IC50 = 10780 nM T55610 CER10L 145969187 IC50 = 1430 nM T55610 CI7X0C 145969829 IC50 = 3040 nM T55610 CEQ31G 145969857 IC50 = 2040 nM T55610 C8G5IP 145972492 IC50 = 5250 nM T55610 CW7T0V 145972540 IC50 = 600 nM T55610 C0ZAH6 145972777 IC50 = 11680 nM T55610 CVY9M5 145972794 IC50 = 5280 nM T55610 COJN36 145974017 IC50 > 15000 nM T55610 C8PHF4 145974424 IC50 = 8740 nM T55610 C9SD7A 145974431 IC50 > 15000 nM T55610 C2H5EC 145974853 IC50 = 2060 nM T55610 CN5R2U 145975516 IC50 = 6520 nM T55610 C6PIW7 145976237 IC50 = 2590 nM T55610 CYS5K7 145976645 IC50 = 8880 nM T55610 CWN92X 145977016 IC50 = 7350 nM T55610 C7HE3Z 145977970 IC50 = 6850 nM T55610 C5R1NG 151545299 IC50 = 4560 nM T55610 CY6S1E 152403353 IC50 = 13800 nM T55610 C64WBL 152584730 IC50 = 11610 nM T55610 CF8Z3X 155510731 IC50 = 22.8 nM T55610 CR68AW 155511636 IC50 = 18100 nM T55610 CSF1T7 155512479 IC50 = 40000 nM T55610 CCL38F 155512808 IC50 = 4000 nM T55610 CLA9C0 155512862 IC50 > 100000 nM T55610 CS38WQ 155513519 IC50 = 37800 nM T55610 C0ZJQ3 155514481 IC50 > 100000 nM T55610 CXTV54 155514795 IC50 = 1600 nM T55610 C2DRJ3 155514884 IC50 = 27400 nM T55610 CX6H5A 155515249 IC50 = 21100 nM T55610 C0DVG8 155517034 IC50 = 40500 nM T55610 CXKH25 155518034 IC50 = 22800 nM T55610 C30IMF 155518712 IC50 > 100000 nM T55610 CP1TH4 155520113 IC50 = 2480 nM T55610 CGU2F7 155520496 IC50 > 100000 nM T55610 CT42DX 155520872 IC50 = 14200 nM T55610 C61KZA 155524227 IC50 = 8900 nM T55610 C1UR2Z 155525413 IC50 = 13200 nM T55610 C6V7SD 155525449 IC50 > 100000 nM T55610 C96WGN 155525554 IC50 > 100000 nM T55610 CXQV24 155526495 IC50 > 100000 nM T55610 C7UDO6 155526802 IC50 = 13300 nM T55610 C8HJY3 155527062 IC50 = 18100 nM T55610 C37LQC 155527106 IC50 = 16700 nM T55610 CP89LD 155527334 IC50 > 100000 nM T55610 CWX8E9 155528670 IC50 > 100000 nM T55610 CD3O0F 155528752 IC50 > 100000 nM T55610 C1E8WZ 155529013 IC50 = 88800 nM T55610 CEV4Z2 155529411 IC50 > 100000 nM T55610 CL3W1J 155529644 IC50 = 10300 nM T55610 CA04QL 155530413 IC50 = 26200 nM T55610 C7PW0Y 155531414 IC50 = 75400 nM T55610 CS9R0Q 155532086 IC50 > 100000 nM T55610 CWG81K 155533235 IC50 > 100000 nM T55610 CCDV47 155533791 IC50 = 4700 nM T55610 CE3Y4L 155533847 IC50 > 100000 nM T55610 CJS5E6 155535208 IC50 = 4240 nM T55610 CP0F5G 155536836 IC50 = 1410 nM T55610 C2GN4P 155538252 IC50 > 100000 nM T55610 CC6Y7R 155539587 IC50 = 10040 nM T55610 CV65ME 155540933 IC50 = 83000 nM T55610 C4NK0M 155541199 IC50 = 7500 nM T55610 C5V6JU 155542174 IC50 = 30300 nM T55610 CK6R3O 155542828 IC50 = 2200 nM T55610 CF5NA0 155545864 IC50 = 8500 nM T55610 CP2Z6H 155546323 IC50 > 100000 nM T55610 C59GSY 155546384 IC50 = 9840 nM T55610 CRI5A9 155547037 IC50 = 9840 nM T55610 CIBK62 155548851 IC50 = 800 nM T55610 C8K2LC 155549309 IC50 = 8530 nM T55610 C87NAR 155549708 IC50 > 100000 nM T55610 C2TML9 155552894 IC50 = 6700 nM T55610 C80OSY 155553753 IC50 > 100000 nM T55610 C7LP8R 155554558 IC50 > 100000 nM T55610 CAB31M 155554811 IC50 = 36900 nM T55610 COP18W 155554892 IC50 > 100000 nM T55610 CY94UD 155556676 IC50 = 930 nM T55610 C6CF8E 155557360 IC50 = 13300 nM T55610 CMB94Q 155557379 IC50 = 1400 nM T55610 CV7A3C 155558225 IC50 = 13200 nM T55610 C73SQD 155558377 IC50 > 100000 nM T55610 C6QT9W 155561428 IC50 = 13300 nM T55610 COZ2V0 155561685 IC50 > 100000 nM T55610 CY3BQ9 155561994 IC50 > 100000 nM T55610 CXTU35 155562845 IC50 = 18100 nM T55610 C0SC5I 155563749 IC50 = 90400 nM T55610 CASY61 155564889 IC50 > 100000 nM T55610 C5STJ2 155565403 IC50 = 10300 nM T55610 C3LD4X 155565589 IC50 = 76400 nM T55610 CN30FA 155566032 IC50 = 2160 nM T55610 CGLV07 155566837 IC50 = 7320 nM T55610 D00REK 5712 IC50 = 1500 nM T55610 D01NUT 5467256 IC50 = 4050 nM T55610 D01OQW 9959532 IC50 = 2600 nM T55610 D04FNI 11657687 IC50 = 100 nM T55610 D05WTI 11550535 IC50 > 30000 nM T55610 D07LUJ 64945 IC50 > 100000 nM T55610 D08VRV 45485203 IC50 = 8320 nM T55610 D09WED 45485202 IC50 = 3170 nM T55610 D0E1ZS 5281297 IC50 = 3510 nM T55610 D0H1WV 45273151 IC50 = 3620 nM T58178 D00ENY 33032 Ki = 1106 nM T58178 D02VKC 3272524 Ki = 13200 nM T58178 D0B0NQ 127894 Ki > 100000 nM T58178 D04XMJ 11249042 Ki > 100000 nM T58178 COC91V 10255 Ki = 32 nM T58178 C37ROZ 439282 Ki = 450 nM T58178 CC0E1V 447081 Ki = 18800 nM T58178 C2BWR8 626468 IC50 = 700 nM T58178 C1EP3D 2733518 Ki > 100000 nM T58178 CWK7X4 4694356 Ki > 100000 nM T58178 CZ63FH 5287393 EC50 = 180000 nM T58178 CZ2SK5 5287396 Ki = 13800 nM T58178 C5Z8VG 6324635 Ki > 10000 nM T58178 C2L6EK 9807075 Ki = 1400 nM T58178 CU09JR 9837067 Ki = 1456 nM T58178 C9TLQ4 9861035 Ki = 3859 nM T58178 CFV03Y 9926589 Ki = 236000 nM T58178 CG0WB9 9958244 Ki = 4100 nM T58178 CLG54O 9977288 IC50 > 50000 nM T58178 CFK0R5 10091990 IC50 > 10000 nM T58178 C7Q1MJ 10132082 IC50 = 62000 nM T58178 CRJ2T0 10219992 EC50 > 100000 nM T58178 CXJP17 10266964 Ki = 107.8 nM T58178 C5PD0H 10330442 Ki = 82500 nM T58178 CJ24TX 10330885 Ki > 100000 nM T58178 CFKJ76 10352480 Ki > 100000 nM T58178 CI1NC2 10379406 Ki = 41.1 nM T58178 C7GIJ3 10398361 Ki = 207000 nM T58178 C1N2VM 10420002 Ki > 1000000 nM T58178 CX1V3L 10437436 Ki = 610 nM T58178 CAQ65T 10494266 Ki = 1404 nM T58178 C1BP3S 10494920 Ki = 27280 nM T58178 CM8JX3 10497847 Ki = 275.3 nM T58178 CL64KJ 10498120 Ki = 90.6 nM T58178 CW1DB8 10515815 Ki > 10000 nM T58178 CA1H6P 10518677 Ki = 27532 nM T58178 C95GPF 10520393 Ki = 288 nM T58178 C6XV7F 10520545 Ki = 1568 nM T58178 CBQ5U4 10522010 Ki > 10000 nM T58178 C91WYV 10524733 Ki = 126.2 nM T58178 CN7ET5 10536623 Ki = 22529 nM T58178 CXE7F5 10541731 Ki = 48 nM T58178 CY53HR 10543350 Ki = 2303.3 nM T58178 CCP30F 10543516 Ki = 146.8 nM T58178 CFRX68 10545609 Ki = 146.6 nM T58178 CQ9UA8 10546918 Ki = 209.6 nM T58178 CPR42C 10559986 Ki = 5373 nM T58178 CY1X4U 10566652 Ki = 54.3 nM T58178 CG8NF3 10566879 Ki = 31.7 nM T58178 C4TS7W 10585396 Ki = 68547 nM T58178 CK20MI 10588564 Ki = 500 nM T58178 CX1J3W 10588885 Ki = 559 nM T58178 CH8R2Z 10589792 Ki = 22340 nM T58178 C71YFN 10592589 Ki = 43929 nM T58178 CKF76J 10592607 Ki = 145.6 nM T58178 CUZ51L 10592608 Ki = 262.7 nM T58178 CO0FS2 10596851 Ki = 667 nM T58178 C4H0FC 10597645 Ki = 129.3 nM T58178 C4BQ9F 10608628 Ki = 10247 nM T58178 C43WUY 10614515 Ki = 93.5 nM T58178 CUN7I9 10632449 Ki = 2984 nM T58178 CQ53LW 10638626 Ki = 6024 nM T58178 CW4A5Q 10660003 Ki = 6969 nM T58178 C5TQN4 10663146 Ki = 131.5 nM T58178 CEA76S 10672549 Ki = 2423.3 nM T58178 C46KUE 10680281 Ki = 41152 nM T58178 C4QB9N 10683926 Ki > 10000 nM T58178 CK9U5T 10685849 Ki = 82.2 nM T58178 CXQ6V2 10689269 Ki = 130.6 nM T58178 C12RGF 10694271 Ki = 1295.7 nM T58178 CBNR83 10708836 Ki = 38.4 nM T58178 CWTN04 10732079 Ki = 4491 nM T58178 C7N5AW 10732793 Ki = 1132 nM T58178 CMQZ05 10733581 Ki = 3845 nM T58178 CQ42JY 10741044 Ki = 1284 nM T58178 C1TRI8 10751988 Ki = 7207 nM T58178 C8AD1O 10754863 Ki = 29.8 nM T58178 C6A4QO 10758246 Ki = 13949 nM T58178 C2EJ0G 10760378 Ki = 3109.2 nM T58178 CLYT96 10767237 Ki > 10000 nM T58178 CASX36 10773867 Ki = 823 nM T58178 CO0B4H 10774436 Ki = 3258 nM T58178 C6U3FQ 10775370 Ki = 2893 nM T58178 CCOE52 10777807 Ki = 1000 nM T58178 CXWT28 10777943 Ki = 339 nM T58178 C7CA4P 10778899 Ki = 4375 nM T58178 C92QWY 10780042 Ki = 6349 nM T58178 C30UTV 10797596 Ki = 160 nM T58178 CXD2H3 10804393 Ki = 169.3 nM T58178 C6KV9E 10804508 Ki = 57.4 nM T58178 CMUE34 10805132 Ki = 4366 nM T58178 CB7R3C 10806437 Ki = 3987 nM T58178 CFOK95 10809478 Ki = 663.3 nM T58178 CZ6AH1 10827292 Ki = 122.5 nM T58178 C4XFQ3 10831138 Ki = 7216 nM T58178 CQA6D3 10846340 Ki = 42809 nM T58178 C4G9SI 10854556 Ki = 5650 nM T58178 CR5XS2 11153198 Ki > 100000 nM T58178 CRS35K 11154806 Ki > 100000 nM T58178 CA83CR 11199813 Ki > 100000 nM T58178 CQ38WM 11219775 Ki > 100000 nM T58178 CGRT02 11288627 Ki > 100000 nM T58178 C8V4UC 11544633 IC50 > 100000 nM T58178 C3NV6L 11742032 IC50 = 37000 nM T58178 C7SHB1 11745400 Ki = 2450 nM T58178 C06UPV 11791928 Ki = 11185 nM T58178 CHUX80 11818375 Ki > 100000 nM T58178 CDGZ79 11820131 Ki > 500000 nM T58178 CM9WF2 15347043 Ki = 2500 nM T58178 C6AYD8 15347044 Ki = 18000 nM T58178 C7ES3B 15839907 Ki = 1580 nM T58178 CYE1O2 18395300 Ki = 46300 nM T58178 CUP4K1 18944678 IC50 = 6700 nM T58178 CLRK62 22097088 Ki = 3900 nM T58178 C0YK6J 22100077 Ki = 28000 nM T58178 CM9D7U 22100122 Ki = 3600 nM T58178 CJ8UB0 22100152 Ki = 1500 nM T58178 CIG65E 22449297 Ki = 5800 nM T58178 C0F8KD 44296355 Ki = 87600 nM T58178 CY4KI5 44296375 Ki = 634000 nM T58178 C0WZ7J 44296493 Ki > 100000 nM T58178 C7JD6F 44296494 Ki > 100000 nM T58178 C0Y8NC 44296575 Ki > 100000 nM T58178 CI9XM2 44296576 Ki = 125000 nM T58178 C6KCR4 44296585 Ki > 100000 nM T58178 CX6LM7 44296601 Ki = 205000 nM T58178 C5LVR2 44296602 Ki > 400000 nM T58178 CJA8X0 44296603 Ki > 10000 nM T58178 CPU32O 44296615 Ki = 193000 nM T58178 CQR8P3 44296800 Ki = 57200 nM T58178 C2VGB7 44296807 Ki > 100010 nM T58178 C1JV4N 44296812 Ki = 255000 nM T58178 C1RIO8 44296822 Ki = 16300 nM T58178 CH3W0P 44301844 Ki = 8250 nM T58178 CJ5X0B 44307207 Ki = 6200 nM T58178 C1JC7K 44307264 Ki = 1200 nM T58178 C8U2SF 44307281 Ki = 23000 nM T58178 CX8AL2 56945410 IC50 > 100000 nM T58178 C0J8AZ 76321095 IC50 = 10000 nM T58178 C0B4KR 76331981 IC50 = 6000 nM T58178 CJ56PL 135423312 IC50 > 30000 nM T58178 D01BAG 16125102 IC50 > 100000 nM T58178 D03NDD 9935648 Ki = 50 nM T58178 D03RGP 1221 Ki > 100000 nM T58178 D09VYB 6420161 IC50 > 300000 nM T58178 D0B2VW 95883 Ki = 10 nM T58178 D0K5UI 6420160 IC50 > 100000 nM T58178 D0K6AF 9839436 Ki = 1.2 nM T58178 D0N1CL 9799478 IC50 = 28000 nM T58178 D0T1MK 656723 Ki > 100000 nM T58178 D0T5SU 158397 Ki > 1000000 nM T34997 D09ZZW 503536 IC50 = 1500 nM T34997 C6IQV0 482174 IC50 = 5700 nM T34997 CY61LO 487910 IC50 = 1700 nM T34997 C6K5JV 487911 IC50 = 16000 nM T34997 C3J5VH 487912 IC50 = 1000 nM T34997 CZNK70 487918 IC50 = 330 nM T34997 CDN3F2 487919 IC50 = 1630 nM T34997 CT76XW 487920 IC50 = 2100 nM T34997 CVA82G 487921 IC50 = 460 nM T34997 CBR46W 487922 IC50 = 1400 nM T34997 CAJ64Q 490750 IC50 < 1000 nM T34997 CMO49H 491114 IC50 = 4300 nM T34997 COB17R 492544 IC50 > 50000 nM T34997 C68MZE 492548 IC50 > 100000 nM T34997 C4JO9E 492549 IC50 = 3280 nM T34997 C1JEY2 492550 IC50 = 300 nM T34997 CRML27 492552 IC50 = 380 nM T34997 C84QRW 493418 IC50 = 5700 nM T34997 CY1WF7 497453 IC50 = 3000 nM T34997 C43PXV 503499 IC50 = 2400 nM T34997 C2BSI5 503516 IC50 = 14000 nM T34997 CFRT87 503517 IC50 = 5400 nM T34997 C3JB0U 503520 IC50 = 13000 nM T34997 CA72XJ 503521 IC50 = 5200 nM T34997 CF14KO 503522 IC50 = 7400 nM T34997 CH18YP 503523 IC50 = 4600 nM T34997 CG6T1D 503524 IC50 = 4100 nM T34997 CLY7T8 503525 IC50 = 750 nM T34997 C37MIA 503526 IC50 = 1000 nM T34997 C8U2AD 503527 IC50 = 12000 nM T34997 CO6R4G 503528 IC50 = 2000 nM T34997 CHA5F8 503529 IC50 > 50000 nM T34997 C41DVG 503530 IC50 = 21000 nM T34997 C5XRJ6 503531 IC50 = 1200 nM T34997 CI1V6W 503532 IC50 > 50000 nM T34997 C84DXH 503533 IC50 = 1400 nM T34997 C7R3CM 503534 IC50 = 2000 nM T34997 CCMU16 503535 IC50 = 3000 nM T34997 C1E4IO 504181 IC50 = 2700 nM T34997 CEJ6U1 504182 IC50 = 1800 nM T34997 CZDS90 504183 IC50 = 1600 nM T34997 C04ONL 504184 IC50 = 2200 nM T34997 C65XPH 504185 IC50 = 11000 nM T34997 CRZN68 504186 IC50 = 42000 nM T34997 CK8CA2 504187 IC50 > 60000 nM T34997 C01MYV 504188 IC50 = 5800 nM T34997 C4C5WD 504189 IC50 = 4300 nM T34997 CIB52E 504190 IC50 = 230 nM T34997 CQ6L1G 504191 IC50 = 12000 nM T34997 C4CW5A 504192 IC50 > 60000 nM T34997 C09ACU 504193 IC50 > 60000 nM T34997 C7T0AD 504194 IC50 = 1300 nM T34997 C7VZY1 504195 IC50 > 60000 nM T34997 CU4EK0 504196 IC50 = 3600 nM T34997 COUS53 504197 IC50 = 5300 nM T34997 CTE3B4 504198 IC50 = 7700 nM T34997 CT81MP 504676 IC50 = 3500 nM T34997 C9FI5K 504680 IC50 = 10600 nM T34997 C8IFN4 504681 IC50 = 31000 nM T34997 CV6OY3 506523 IC50 = 1400 nM T34997 CQX7S4 506524 IC50 = 390 nM T34997 CXD73I 506525 IC50 = 1800 nM T34997 C6ANI5 506528 IC50 = 9000 nM T34997 CRU30I 507613 IC50 = 900 nM T34997 CI8SQ4 511361 IC50 > 50000 nM T34997 C02LPN 511362 IC50 = 30000 nM T34997 CJIW67 511363 IC50 = 13000 nM T34997 C3KG1M 511364 IC50 = 43000 nM T34997 CU85HK 511365 IC50 = 10700 nM T34997 C20EKN 511366 IC50 = 5900 nM T34997 C3FX8J 511367 IC50 = 31000 nM T34997 C4DEY1 511368 IC50 = 3700 nM T34997 CC2J9M 511369 IC50 = 5600 nM T34997 CIU5M2 511370 IC50 = 11000 nM T34997 C5CG4I 511371 IC50 = 5000 nM T34997 CTO87P 511372 IC50 = 2700 nM T34997 C5BJ6S 511373 IC50 = 26000 nM T34997 CDWB40 511374 IC50 = 15000 nM T34997 CDH29C 511375 IC50 = 31000 nM T34997 C8ZJD7 511376 IC50 = 31000 nM T34997 CJ56OH 513150 IC50 < 10000 nM T34997 C5BN4U 513891 IC50 = 12000 nM T34997 CVI54C 657065 IC50 = 1200 nM T34997 CUC54L 3008068 IC50 = 5000 nM T34997 CJ5NO6 3008069 IC50 = 34000 nM T34997 CQO9Y3 3008070 IC50 > 32000 nM T34997 CXM1K9 3008071 IC50 > 50000 nM T34997 CJ2NY3 3008418 IC50 = 20000 nM T34997 CIJ2T0 3008419 IC50 > 50000 nM T34997 CWD1X0 3008420 IC50 = 14000 nM T34997 C4K2JP 3008421 IC50 > 50000 nM T34997 CAN83S 3008422 IC50 = 13000 nM T34997 CMDQ27 4468931 IC50 = 1800 nM T34997 CK9WY1 5278824 IC50 = 100 nM T34997 C5MEQ4 5278825 IC50 = 110 nM T34997 C1F0AN 5278826 IC50 = 45 nM T34997 CV0O6S 5482516 IC50 = 15600 nM T34997 CEM30Z 5483089 IC50 = 8900 nM T34997 CJL21S 9853197 IC50 = 60 nM T34997 CJW4M9 9917616 IC50 = 11000 nM T34997 C39ZBC 10207572 IC50 = 30000 nM T34997 CGA86Z 10259200 IC50 = 12000 nM T34997 CJ46UK 10439772 IC50 = 420 nM T34997 COM8C5 21148125 IC50 = 16000 nM T34997 C1TW3V 22209806 IC50 > 50000 nM T34997 C8GVX3 22209808 IC50 > 50000 nM T34997 C6AS7E 22209811 IC50 = 3300 nM T34997 CLW13P 22209812 IC50 = 1700 nM T34997 C1TA6Z 22209813 IC50 = 440 nM T34997 CGUC83 22210989 IC50 = 58000 nM T34997 CV97ER 22210996 IC50 = 18000 nM T34997 C2BA1K 22211000 IC50 = 27000 nM T34997 C78AKX 22211010 IC50 > 100000 nM T34997 CL7M9B 22211011 IC50 = 32000 nM T34997 C1L8TE 22211012 IC50 = 18000 nM T34997 C0NYS5 22211016 IC50 = 50000 nM T34997 C67QJW 22211018 IC50 > 100000 nM T34997 CV9S2O 22211019 IC50 = 13000 nM T34997 C4UB6Q 22211020 IC50 = 14000 nM T34997 CBUV46 22211021 IC50 = 62000 nM T34997 CS9B7N 22211022 IC50 > 100000 nM T34997 CK81WO 25078062 IC50 = 3400 nM T34997 CYDW71 44268661 IC50 > 60000 nM T34997 C6S3AT 44268682 IC50 > 60000 nM T34997 CDJ0X4 44308299 IC50 > 100000 nM T34997 CIO1C2 44308345 IC50 > 100000 nM T34997 CX14BI 44308422 IC50 > 100000 nM T34997 CE3PS8 44308752 IC50 = 34000 nM T34997 CK2P5O 44375061 IC50 > 50000 nM T34997 C4CVW1 44375110 IC50 > 50000 nM T34997 C72KUL 44375154 IC50 = 9400 nM T34997 C1SBO9 44375192 IC50 > 50000 nM T34997 C42GUE 44375229 IC50 = 5300 nM T34997 CX76FI 44388198 IC50 = 350 nM T34997 CVW6O4 44399745 IC50 = 79432.82 nM T34997 CDRP83 44399750 IC50 = 50118.72 nM T34997 CW6NY8 44399751 IC50 = 5011.87 nM T34997 CM5W8Q 44399752 IC50 = 6309.57 nM T34997 C34WSP 44399753 IC50 = 10000 nM T34997 CE0T1O 44399754 IC50 = 1995.26 nM T34997 CT86CR 44399784 IC50 = 25118.86 nM T34997 C6GWS9 44399837 IC50 = 31622.78 nM T34997 C4AI1T 44399861 IC50 = 100000 nM T34997 CTX79F 44399866 IC50 = 25118.86 nM T34997 CP4KB7 44399867 IC50 = 794.33 nM T34997 C0WRU5 44399868 IC50 = 15848.93 nM T34997 C8JP2A 44399889 IC50 = 50118.72 nM T34997 CO4H3V 44399938 IC50 = 10000 nM T34997 CYH7F9 44399975 IC50 = 6309.57 nM T34997 CZRF38 44399976 IC50 = 6309.57 nM T34997 CATH48 44399977 IC50 = 6309.57 nM T34997 CL9NS3 44399978 IC50 > 199526.23 nM T34997 C9YO4K 44399979 IC50 > 199526.23 nM T34997 CX8M3O 44400003 IC50 = 39810.72 nM T34997 C4X1OG 44400004 IC50 = 19952.62 nM T34997 C5EV1S 44400005 IC50 = 158489.32 nM T34997 CFRU27 44400006 IC50 = 199526.23 nM T34997 C7FO3T 44400007 IC50 = 251188.64 nM T34997 CA6P2U 44400008 IC50 = 100000 nM T34997 CQP47M 44400009 IC50 = 7943.28 nM T34997 CCRB97 44400010 IC50 = 3981.07 nM T34997 CT40SR 44400033 IC50 = 31622.78 nM T34997 CA96HO 44400076 IC50 > 1000000 nM T34997 CX7O2Z 44400112 IC50 > 199526.23 nM T34997 C6Z5NC 44400113 IC50 > 199526.23 nM T34997 C6PCE5 44400114 IC50 = 31622.78 nM T34997 C95CRD 44400115 IC50 = 19952.62 nM T34997 CW5G3Z 73347065 IC50 > 50000 nM T34997 C6TNQ8 135412361 IC50 = 800 nM T34997 C53AWL 135434400 IC50 = 100 nM T83979 D04EEU 53001 IC50 > 100000 nM T83979 D09QRO 55390 IC50 = 100000 nM T83979 D0OO6A 5284442 IC50 > 100000 nM T83979 CF06EN 795 IC50 = 4000000 nM T83979 C7I6HX 53555 IC50 > 100000 nM T83979 CFJ3L6 13094289 IC50 > 100000 nM T83979 CQ8L5Y 13569173 IC50 > 100000 nM T83979 CLOP75 13569178 IC50 > 1000000 nM T83979 C4BT5G 13569185 IC50 > 1000000 nM T83979 C1VNT2 13569189 IC50 > 100000 nM T83979 CE01PH 13569191 IC50 > 100000 nM T83979 CC07NV 13569194 IC50 > 100000 nM T83979 C37HVK 13569196 IC50 > 100000 nM T83979 C4GRJ1 13569197 IC50 > 100000 nM T83979 CCB9W8 13569199 IC50 > 1000000 nM T83979 CCAN10 13594154 IC50 > 100000 nM T83979 CCF4E0 13594155 IC50 > 100000 nM T83979 C4GR2M 13594156 IC50 > 100000 nM T83979 C5EI9O 13594158 IC50 > 100000 nM T83979 CB94PC 13594159 IC50 > 100000 nM T83979 C39EWI 13594160 IC50 > 100000 nM T83979 C3NV6O 13594161 IC50 > 100000 nM T83979 C61EUC 13594162 IC50 > 100000 nM T83979 C4CIL0 13594163 IC50 > 100000 nM T83979 CLA7H9 13663090 IC50 > 10 nM T83979 CBL5S7 13663091 IC50 > 100000 nM T83979 C2Y5SB 13663093 IC50 > 100000 nM T83979 C2A5FS 13663094 IC50 > 100000 nM T83979 C6XU4Y 13663096 IC50 > 100000 nM T83979 CPFG92 13663097 IC50 > 100000 nM T83979 CU6RA8 44209341 IC50 = 75000 nM T83979 C7RS8L 44209342 IC50 > 100000 nM T83979 CO53TB 44209343 IC50 < 1000 nM T83979 CC79FZ 44209484 IC50 = 28000 nM T83979 CZE9V1 44209485 IC50 > 100000 nM T83979 C3FWQ1 44209486 IC50 = 12000 nM T83979 CX73JP 44343361 IC50 > 100000 nM T83979 CFG3R2 44374426 IC50 = 37000 nM T83979 CU8K1E 44374438 IC50 = 9000 nM T83979 CKW29G 44374442 IC50 = 60000 nM T83979 C0LHQ3 44374492 IC50 = 9000 nM T83979 C8LI5R 44374505 IC50 = 32000 nM T83979 CU4N0J 44374506 IC50 = 4000 nM T83979 C2H0XN 44374508 IC50 > 100000 nM T83979 C09MVC 44374535 IC50 = 2000 nM T83979 C6TDS3 44374545 IC50 = 2000 nM T83979 C5Q9XG 44374548 IC50 = 3000 nM T83979 CDG36Y 44374549 IC50 < 1000 nM T83979 C4CG0B 44374558 IC50 = 7000 nM T83979 C43AFG 44374559 IC50 = 14000 nM T83979 CP4XW7 44374560 IC50 = 13000 nM T83979 C0AYJ4 44374685 IC50 = 7000 nM T83979 C1ZOS4 44374692 IC50 = 25000 nM T83979 C2YT1N 44374696 IC50 = 2500 nM T83979 C6ZQ3E 44374697 IC50 = 2000 nM T83979 C0UOT1 44374698 IC50 = 8000 nM T83979 C7BDM5 44374700 IC50 > 100000 nM T83979 CWU80E 44374721 IC50 = 13000 nM T83979 C9I4ZT 44374740 IC50 = 23000 nM T83979 CK1A0I 44374752 IC50 = 73000 nM T83979 CO8Q1T 44374930 IC50 > 100000 nM T83979 C07GQT 44374931 IC50 = 4000 nM T83979 CT8EZ5 44374945 IC50 = 5000 nM T83979 CMC19F 44374965 IC50 > 100000 nM T83979 C7O3UE 44374966 IC50 = 51000 nM T83979 C9MJA1 44374981 IC50 < 1000 nM T83979 C79GUZ 44374982 IC50 = 40000 nM T83979 C3IXM4 54728414 IC50 > 100000 nM T83979 D00RRV 792486 IC50 = 650000 nM T83979 D01CGR 194468 IC50 > 100000 nM T83979 D0R8NE 13569172 IC50 > 1000000 nM T83979 D0Y1YZ 13569177 IC50 > 100000 nM T63083 C95TRU 720237 IC50 = 17850 nM T63083 CO8G9N 779728 IC50 = 38170 nM T63083 C46XHS 796318 IC50 = 19700 nM T63083 CPB83T 1049183 IC50 = 14880 nM T63083 CBO6D7 1074953 IC50 = 6820 nM T63083 COW3Q9 1180676 IC50 = 6430 nM T63083 C73KAQ 1661927 IC50 = 8320 nM T63083 C8IAL0 2814482 IC50 = 13100 nM T63083 CRGD04 3300756 EC50 = 50000 nM T63083 CIE0C3 3301542 EC50 = 16000 nM T63083 C58JVK 3513680 EC50 = 16000 nM T63083 CYAQ75 3909954 EC50 = 38000 nM T63083 CHFT32 4245983 EC50 = 10000 nM T63083 CI4KB3 4246127 EC50 = 18400 nM T63083 C9YM4Z 5738263 IC50 = 6000 nM T63083 C12LCY 18553874 EC50 = 53000 nM T63083 C93ZUL 41026155 EC50 = 95000 nM T63083 CY7KZ2 44422142 IC50 > 100000 nM T63083 C7NZY5 46899803 IC50 = 2700 nM T63083 CTD10P 46899807 Ki = 750 nM T63083 CTQ19B 46919033 IC50 = 2100 nM T63083 CWEX47 49864240 IC50 = 3500 nM T63083 CTJA37 49864241 IC50 > 100000 nM T63083 CEZ17W 49864242 IC50 = 6000 nM T63083 C0MP6Y 49864243 IC50 > 40000 nM T63083 C2WGE8 49864244 Ki > 40000 nM T63083 C8S3NX 49864245 Ki = 1800 nM T63083 CH1D4F 49864246 Ki = 4200 nM T63083 C2SHP9 60148051 IC50 = 71700 nM T63083 CVR30K 60148052 IC50 = 79400 nM T63083 CB0WP2 71544709 IC50 > 50000 nM T63083 CXM8T1 71544714 IC50 = 370 nM T63083 CQH43A 71544715 IC50 = 250 nM T63083 C1PM7R 71546685 IC50 = 13160 nM T63083 C2UL1O 71546686 IC50 = 7910 nM T63083 C1BX4E 71546836 IC50 = 9940 nM T63083 C6JQK3 71546837 IC50 = 3100 nM T63083 CL2ZK1 71546989 IC50 = 5290 nM T63083 CTQH17 71546991 IC50 = 15620 nM T63083 CHX0O9 71546992 IC50 = 2140 nM T63083 C3H7AG 71546993 IC50 = 1400 nM T63083 CS0U6O 71547136 IC50 = 930 nM T63083 C69OMQ 71547137 IC50 = 810 nM T63083 C5H8UR 71547138 IC50 = 44170 nM T63083 CAK0G8 71547140 IC50 > 50000 nM T63083 CZ8A4H 127048228 IC50 = 27600 nM T63083 CA82DT 127048584 IC50 = 13200 nM T63083 C02LUY 127049243 IC50 = 64900 nM T63083 CYH4Q3 127049901 IC50 > 100000 nM T63083 CCU43I 127050093 IC50 > 100000 nM T63083 C4IJE3 127050408 IC50 = 81500 nM T63083 C6CVX2 127050409 IC50 > 100000 nM T63083 CTI62A 127050410 IC50 = 34000 nM T63083 C8A5DF 127050411 IC50 > 100000 nM T63083 C8T0BU 127050412 IC50 = 38600 nM T63083 C4ON3T 127050413 IC50 = 46100 nM T63083 CC3H0K 127050490 IC50 > 100000 nM T63083 C47DNF 127050498 IC50 > 100000 nM T63083 C3A8YK 127051390 IC50 = 8400 nM T63083 C7YV3Q 127052027 IC50 = 27200 nM T63083 C0SR6Z 127052037 IC50 > 100000 nM T63083 CW1GF2 127052549 IC50 = 13000 nM T63083 C7MI0X 127052564 IC50 = 91100 nM T63083 CX80QY 127052565 IC50 > 100000 nM T63083 C0UDH3 127052566 IC50 = 22100 nM T63083 C70JDH 127052567 IC50 = 3000 nM T63083 CLR8E9 127052568 IC50 > 100000 nM T63083 C0Q5JZ 127052644 IC50 = 57800 nM T63083 CLFY78 127052833 IC50 = 9800 nM T63083 CV8C0Z 127052854 IC50 = 20000 nM T63083 CTF12X 131953896 EC50 = 25000 nM T63083 CE2L6C 136084728 EC50 = 8000 nM T63083 CR9Q1W 136084730 EC50 = 34000 nM T63083 CUX8D4 136094853 IC50 > 100000 nM T63083 CSO0M3 136219342 EC50 = 29000 nM T63083 CKF5O0 136244146 EC50 = 59000 nM T63083 CJW20N 137225003 IC50 = 27600 nM T63083 CT1PR6 137225029 IC50 = 35000 nM T63083 C3RCM0 155510948 EC50 = 40000 nM T63083 CL2BJ6 155512370 EC50 = 25000 nM T63083 CL8QU5 155517576 EC50 = 19000 nM T63083 C46KRC 155517883 EC50 = 28000 nM T63083 CI0FA9 155528805 EC50 = 20000 nM T63083 CURJ89 155530004 EC50 = 70000 nM T63083 C8ZB4J 155533293 EC50 = 2000 nM T63083 C74NLT 155534052 EC50 = 10000 nM T63083 C8Z4VT 155540192 EC50 = 950 nM T63083 C06PEO 155546192 EC50 = 8000 nM T63083 CGU0O5 155547239 EC50 = 70000 nM T63083 C0S1YP 155547558 EC50 = 18000 nM T63083 C03QHV 155549243 EC50 = 20000 nM T63083 CP73ZA 155549425 EC50 = 33000 nM T63083 CCU87L 155549847 EC50 = 42000 nM T63083 C0VFR1 155555558 EC50 = 100000 nM T63083 CAOM03 155556006 EC50 = 90000 nM T63083 CX79JY 155557552 EC50 = 24000 nM T63083 C1AS5N 155557802 EC50 = 50000 nM T63083 C9EJ2N 155561532 EC50 = 46000 nM T63083 C24KCL 155563759 EC50 = 15000 nM T63083 CZTD74 155564150 EC50 = 13000 nM T63083 CYF1R3 155565633 EC50 = 15000 nM T63083 CXK60A 155567395 EC50 = 45000 nM T63083 C19ANC 155567965 EC50 = 17000 nM T63083 CYH84F 155569452 EC50 = 65000 nM T42881 C9KP5F 7518 IC50 = 9000 nM T42881 C7HM4W 69914 IC50 > 34000 nM T42881 C6I4RP 456164 IC50 > 300000 nM T42881 C19DBJ 475734 IC50 = 19000 nM T42881 CN91BS 477469 IC50 = 800 nM T42881 C0M7DF 477470 IC50 = 3500 nM T42881 CP9LE1 477471 IC50 = 19 nM T42881 CGTR95 477472 IC50 = 14 nM T42881 CJ0ID1 477473 IC50 = 1100 nM T42881 C1TUN0 477474 IC50 = 940 nM T42881 C2LGM8 477475 IC50 = 1000 nM T42881 C0K8ET 477476 IC50 = 1100 nM T42881 CI8M7V 477477 IC50 = 1400 nM T42881 C9EK8I 477478 IC50 = 1500 nM T42881 C3B1HT 477479 IC50 = 45 nM T42881 CPG67H 477480 IC50 = 61 nM T42881 CWU1M8 477481 IC50 = 3800 nM T42881 CUP20R 477482 IC50 = 2400 nM T42881 CQ28ZD 477483 IC50 = 2200 nM T42881 CB8VG0 477484 IC50 = 55 nM T42881 C4UVT0 477485 IC50 > 33000 nM T42881 C5K6AW 477486 IC50 > 33000 nM T42881 CDS0V1 477487 IC50 = 2000 nM T42881 CQEH07 477488 IC50 = 3700 nM T42881 C4F8OW 477489 IC50 = 11000 nM T42881 C2EJG6 478959 IC50 = 6500 nM T42881 C8FQ5N 478963 IC50 > 100000 nM T42881 C61JON 478964 IC50 > 100000 nM T42881 CT26XP 478965 IC50 = 68000 nM T42881 C4CD1L 478966 IC50 = 42000 nM T42881 CSLD96 478967 IC50 > 100000 nM T42881 CMT6C7 478968 IC50 > 100000 nM T42881 CO30YD 478969 IC50 = 27000 nM T42881 CK40HJ 478970 IC50 > 100000 nM T42881 C4G1UL 478971 IC50 = 86000 nM T42881 C6P7EJ 478972 IC50 = 100000 nM T42881 CM4Z2U 478973 IC50 > 100000 nM T42881 C6SC2U 478974 IC50 > 100000 nM T42881 CQS5M3 478975 IC50 > 100000 nM T42881 C3AYB0 479059 IC50 = 20000 nM T42881 CL2A5E 479060 IC50 > 100000 nM T42881 CO0V3F 479061 IC50 = 50000 nM T42881 C9EAL6 482277 IC50 = 1300 nM T42881 C58PLQ 482278 IC50 = 1400 nM T42881 C2G9IH 482279 IC50 = 300 nM T42881 C5L4ED 482280 IC50 = 400 nM T42881 CTW1J9 482282 IC50 = 1900 nM T42881 CK0O9U 482283 IC50 = 2400 nM T42881 CX0SQ5 482284 IC50 = 6500 nM T42881 C6Y5SA 482285 IC50 = 2100 nM T42881 C2D7MH 482286 IC50 = 2000 nM T42881 CAZV26 482287 IC50 = 2500 nM T42881 C2QP9I 482288 IC50 = 1000 nM T42881 C3L9TI 482289 IC50 = 75000 nM T42881 CO3N0A 482290 IC50 = 1200 nM T42881 CZ15KR 482291 IC50 = 6400 nM T42881 C0HV7G 482292 IC50 = 3600 nM T42881 CFL1P5 490579 IC50 = 110000 nM T42881 C5K8FZ 490581 IC50 = 40000 nM T42881 C07BSR 490582 IC50 = 13000 nM T42881 CLQ15W 490585 IC50 > 500000 nM T42881 C8X5TQ 490588 IC50 = 9000 nM T42881 CW2C3Z 490589 IC50 = 16000 nM T42881 C7IOC8 490590 IC50 = 72000 nM T42881 CRB0A1 490592 IC50 > 500000 nM T42881 CLWX67 490599 IC50 > 500000 nM T42881 C13NET 490601 IC50 ~ 500000 nM T42881 CIK65R 490618 IC50 = 1400 nM T42881 C5NQC4 490619 IC50 = 2200 nM T42881 C85PJN 493455 IC50 > 500000 nM T42881 CD5H1W 493456 IC50 = 148000 nM T42881 C4WL2A 493458 IC50 > 500000 nM T42881 CYB9U0 493459 IC50 = 250000 nM T42881 CMO83V 493460 IC50 ~ 500000 nM T42881 CWB35S 493461 IC50 ~ 500000 nM T42881 C2LQ3J 493462 IC50 = 1400 nM T42881 CG8ZF1 493463 IC50 = 5100 nM T42881 C4K7TP 493464 IC50 > 100000 nM T42881 CBE06W 493465 IC50 = 22000 nM T42881 C8YJE9 493466 IC50 = 6600 nM T42881 CL0C4A 493467 IC50 = 41000 nM T42881 CJ8WU4 493468 IC50 = 2100 nM T42881 C3YWS6 511075 IC50 = 1100 nM T42881 CN42SP 511076 Ki = 60 nM T42881 CW0HA1 511077 Ki = 40 nM T42881 C23MOD 511078 IC50 = 2100 nM T42881 C30XFM 511079 IC50 = 1800 nM T42881 C02TMH 511080 IC50 = 840 nM T42881 C48PWK 511081 Ki = 99 nM T42881 C4WGO9 511082 Ki = 39 nM T42881 CZL3V2 511083 IC50 = 65000 nM T42881 C6OR5W 511084 Ki = 33 nM T42881 C2YWZ0 511085 Ki = 2 nM T42881 CJN6A2 511086 Ki = 21 nM T42881 C69CKY 511087 IC50 = 390 nM T42881 C90CZS 511088 Ki = 79 nM T42881 C9VA3I 511089 IC50 = 890 nM T42881 C15HMK 511090 IC50 = 1400 nM T42881 CMO7R5 511091 Ki = 2 nM T42881 CZ2EM8 511092 Ki = 9 nM T42881 CZDJ38 511093 Ki = 15 nM T42881 CCU7P6 511094 Ki = 18 nM T42881 CS5F2L 511095 Ki = 38 nM T42881 CLDW79 511096 IC50 = 650 nM T42881 CO9D3W 511097 IC50 = 470 nM T42881 CNK95T 511098 IC50 = 590 nM T42881 CLP72B 511099 IC50 = 650 nM T42881 C97CEK 511100 IC50 = 1400 nM T42881 CRKH21 511101 IC50 = 260 nM T42881 CJY90S 511102 IC50 = 840 nM T42881 C7AB3L 511103 IC50 = 1400 nM T42881 CJ1G7C 511104 Ki = 79 nM T42881 CGY4E7 511105 Ki = 33 nM T42881 CGU9L8 511106 Ki = 16 nM T42881 CK61WM 511107 Ki = 9 nM T42881 C13VZH 511108 IC50 > 20000 nM T42881 CKY3N5 511109 IC50 = 8700 nM T42881 CPE4G3 511110 Ki = 446 nM T42881 CT0P5D 511111 Ki = 10 nM T42881 C86QZC 511113 Ki = 0.31 nM T42881 C0Q3EW 511114 IC50 = 1100 nM T42881 CU63JM 511115 IC50 = 290 nM T42881 C5EOW8 511116 IC50 = 240 nM T42881 CPBK80 511117 IC50 = 460 nM T42881 CQ30MA 511118 IC50 = 210 nM T42881 CFH21A 511119 IC50 = 230 nM T42881 CZ1T8B 511120 IC50 = 360 nM T42881 CB1CI2 511121 Ki = 25 nM T42881 CDC14A 511122 Ki = 7.4 nM T42881 CN8GM9 511123 Ki = 20 nM T42881 CRB49E 511124 Ki = 43 nM T42881 CK60YU 511125 Ki = 21 nM T42881 CB9L3K 511126 IC50 = 870 nM T42881 C4G3ED 3008802 IC50 = 15.3 nM T42881 CKFY95 3008803 IC50 = 21.3 nM T42881 CU6T8M 3008804 IC50 = 15.2 nM T42881 CY90XK 3008805 IC50 = 4.8 nM T42881 CV1QT6 3008806 IC50 = 3.1 nM T42881 CW7Y9Q 3008807 IC50 = 2.8 nM T42881 CVQ5K3 3008808 IC50 = 5.1 nM T42881 C1DJZ4 3008809 IC50 = 6.1 nM T42881 CA7R9N 3008810 IC50 = 7.4 nM T42881 C4CM8P 5481492 IC50 = 21000 nM T42881 C1RF9K 6475392 IC50 = 30 nM T42881 C8X1YP 6475393 IC50 = 260 nM T42881 C93ASX 6475394 IC50 = 60 nM T42881 CGE3O4 6475395 IC50 = 29 nM T42881 C3GB4A 6475396 IC50 = 41 nM T42881 C27PRL 6475397 IC50 = 31 nM T42881 C5A2MF 6475398 IC50 = 14 nM T42881 C3CF5L 6475399 IC50 = 29 nM T42881 CLJ32T 6475400 IC50 = 2300 nM T42881 CQ2DL0 6475401 IC50 = 370 nM T42881 CYJ4I8 6476665 Ki = 20 nM T42881 C0Y8DK 6479584 IC50 = 66 nM T42881 CD8VX6 6479585 IC50 = 9.5 nM T42881 C5CUB2 6479586 IC50 = 6.3 nM T42881 CGPO51 6479587 IC50 = 3.4 nM T42881 C2NW6D 6479588 IC50 = 3.7 nM T42881 C4RW8P 6479589 IC50 = 3.2 nM T42881 CUQD91 6479590 IC50 = 15.1 nM T42881 CZ51XM 6479591 IC50 = 3.2 nM T42881 CRJL96 6479592 IC50 = 10.5 nM T42881 CIDB89 6479593 IC50 = 7.5 nM T42881 CSEJ15 6479594 IC50 = 4.3 nM T42881 C69PRI 6479596 IC50 = 6.6 nM T42881 C70QAF 6479597 IC50 = 15 nM T42881 C38CHN 6479598 IC50 > 50 nM T42881 CVB5Y8 6479599 IC50 > 50 nM T42881 C3M1OL 6479600 IC50 > 50 nM T42881 C89RJV 6479601 IC50 > 50 nM T42881 CE1ZT6 6479602 IC50 = 43 nM T42881 CG3DZ0 6479603 IC50 > 50 nM T42881 CH3L2P 6479604 IC50 = 6.7 nM T42881 CH3P1W 6479605 IC50 = 4.7 nM T42881 CMB53F 6479606 IC50 = 8.3 nM T42881 C9B1MT 6479607 IC50 > 50 nM T42881 CI8CH1 6479608 IC50 = 17.4 nM T42881 CPD8N9 6479609 IC50 = 2.7 nM T42881 C24JMD 6479610 IC50 = 6.9 nM T42881 CN1ET7 6479611 IC50 = 6.9 nM T42881 CW8IQ6 6481314 IC50 ~ 500000 nM T42881 CDEX87 10334241 IC50 = 600 nM T42881 CBT7O8 10874917 IC50 > 500000 nM T42881 C0GX9Q 10894271 IC50 = 50000 nM T42881 CRK5G8 11025393 IC50 > 500000 nM T42881 C6BF5A 11037447 IC50 = 159000 nM T42881 C0J4QW 11113965 IC50 = 540 nM T42881 C9ESN4 11129373 IC50 = 1500 nM T42881 CGK0R6 11316755 IC50 = 6.5 nM T42881 CUG78P 15959480 IC50 = 10000 nM T42881 C8D6VK 44282051 IC50 = 70 nM T42881 CBO0A8 44295551 IC50 > 500000 nM T42881 C4GUO2 44295588 IC50 = 7000 nM T42881 CV09FP 44295599 IC50 = 13000 nM T42881 CRQ08J 44295704 IC50 = 11000 nM T42881 C6ENC1 44295724 IC50 > 1000000 nM T42881 CO9D7H 44295747 IC50 = 11500 nM T42881 C7EI6N 44295781 IC50 = 63000 nM T42881 C1PNL3 44295803 IC50 = 45000 nM T42881 CYK49R 44295804 IC50 = 79000 nM T42881 CHT48A 44295910 IC50 > 500000 nM T42881 CJ0N2Y 44295914 IC50 = 14000 nM T42881 CVY24Z 44295929 IC50 = 6000 nM T42881 CU2E8J 44295937 IC50 = 79000 nM T42881 CVQT37 44295946 IC50 > 100000 nM T42881 CJMN58 44295948 IC50 = 5000 nM T42881 CI04EU 44295967 IC50 = 32000 nM T42881 CWEA02 44295973 IC50 = 6000 nM T42881 CZ7OG6 44296004 IC50 = 126000 nM T42881 CST8Q6 44296005 IC50 = 133000 nM T42881 CZ83YK 44296193 IC50 = 10000 nM T42881 C1F4NK 44296194 IC50 = 9000 nM T42881 CX4ZJ8 44296321 IC50 = 398000 nM T42881 C8J0EP 44296322 IC50 > 500000 nM T42881 C1OBL2 44296323 IC50 > 500000 nM T42881 CSG82W 44347283 IC50 = 600 nM T42881 C4VHU9 44347332 IC50 > 34000 nM T42881 C65IDZ 44347333 IC50 = 460 nM T42881 CBN3T4 44347550 IC50 = 1400 nM T42881 CE6U7Z 44347565 IC50 = 60 nM T42881 C17GPK 44347574 IC50 = 100 nM T42881 CG97UR 44347575 IC50 = 200 nM T42881 CQE5J3 44347576 IC50 > 34000 nM T42881 CH27UB 44347588 IC50 = 60 nM T42881 CMSP60 44347589 IC50 = 100 nM T42881 C4Q5SC 44347590 IC50 > 34000 nM T42881 CSAP19 44347600 IC50 = 180 nM T42881 CZO2U6 44347649 IC50 = 180 nM T42881 CK27CA 44347665 IC50 = 100 nM T42881 CA4UR7 44347666 IC50 = 110 nM T42881 C6EYM4 44347667 IC50 > 34000 nM T42881 C7ABL6 44347792 IC50 = 17000 nM T42881 C8CA1M 44347852 IC50 > 100000 nM T42881 CSD7B6 71461709 IC50 = 72000 nM T42881 CO1YX7 71461732 IC50 > 100000 nM T59654 D01ZRI 6450551 IC50 > 10000 nM T59654 D03HUX 49792852 IC50 > 10000 nM T59654 D0E3TC 44259 IC50 = 471 nM T59654 D0O0LQ 11364421 IC50 = 13.55 nM T59654 D0P1CV 46191454 IC50 > 10000 nM T59654 D0T3ME 156422 IC50 > 30000 nM T59654 C3ZVJ9 10281 IC50 = 14720 nM T59654 CIHY32 2190510 IC50 = 1700 nM T59654 CVZ9D0 3162171 IC50 > 10000 nM T59654 C7HBP6 10429593 IC50 > 10000 nM T59654 CE80VT 11656480 IC50 = 21 nM T59654 C5YW7P 24825755 IC50 = 3519 nM T59654 C7PYN2 24971417 IC50 = 1449 nM T59654 CN1D2A 24971422 IC50 = 4 nM T59654 C3LOR9 24971423 IC50 = 172 nM T59654 CQEV29 24992861 IC50 = 2 nM T59654 CCZF80 24992862 IC50 = 12 nM T59654 CU5B6R 24992864 IC50 > 10000 nM T59654 C4EG8R 24993189 IC50 = 238 nM T59654 CNG96H 25210579 IC50 > 10000 nM T59654 C13QXB 44236351 IC50 = 9 nM T59654 C5M8UY 46886877 IC50 = 109 nM T59654 C3RIH2 46886957 IC50 = 261 nM T59654 CMU45C 46886960 IC50 = 24 nM T59654 C7JG4Q 46887069 IC50 = 14 nM T59654 CYG3B2 46887070 IC50 = 27 nM T59654 C82SLV 46887071 IC50 = 509 nM T59654 C1W3QP 46887105 IC50 = 2666 nM T59654 C45OAG 46887187 IC50 = 12 nM T59654 CW13FN 46887188 IC50 = 2104 nM T59654 C5X8BP 46887189 IC50 > 10000 nM T59654 CB8Q1F 46887190 IC50 > 10000 nM T59654 CK1YB8 46887222 IC50 = 82 nM T59654 CBC62W 50899254 IC50 > 10000 nM T59654 C7SR2D 52940661 IC50 = 190 nM T59654 CQVE12 52942317 IC50 = 3415 nM T59654 CISC65 52943186 IC50 = 1280 nM T59654 CKCN74 52943243 IC50 > 10000 nM T59654 C2N5GH 52943310 IC50 = 3387 nM T59654 C0LSU9 52944272 IC50 = 768 nM T59654 CF63AS 52945523 IC50 > 10000 nM T59654 CQ30DI 52945929 IC50 > 10000 nM T59654 CG8HT0 52946706 IC50 > 10000 nM T59654 CQZX58 52946971 IC50 = 429 nM T59654 C84FOX 52946976 IC50 = 762 nM T59654 CRL93S 52947958 IC50 = 206 nM T59654 CP80TO 52947965 IC50 > 10000 nM T59654 C6O7CR 53249964 IC50 = 130 nM T59654 C4RLN7 53252570 IC50 = 1230 nM T59654 C6S1OX 53252617 IC50 = 350 nM T59654 CO09HS 53252703 IC50 = 470 nM T59654 C8MG1N 53253240 IC50 = 6080 nM T59654 CQ1EJ0 53253241 IC50 = 1070 nM T59654 CFS57D 53261787 IC50 = 21 nM T59654 C87LRX 53261846 IC50 = 7 nM T59654 C25YMU 53261848 IC50 = 103 nM T59654 C8NA4L 53384644 IC50 > 30000 nM T59654 C30AQN 54580351 IC50 > 10000 nM T59654 CEC0T9 54581348 IC50 > 10000 nM T59654 CL42MV 54582373 IC50 > 10000 nM T59654 CF7P8Y 54582374 IC50 > 10000 nM T59654 C30RMF 54583357 IC50 = 3855 nM T59654 CKM86O 54583358 IC50 = 1494 nM T59654 CG9LS2 54583359 IC50 = 1499 nM T59654 CY9J3B 54584304 IC50 = 1453 nM T59654 CP2Z0T 54584305 IC50 = 762 nM T59654 CI4SU2 54585267 IC50 = 2254 nM T59654 C51NCQ 54585268 IC50 > 10000 nM T59654 CJ1S9E 54585269 IC50 = 1364 nM T59654 CP86VM 54586220 IC50 > 10000 nM T59654 C8WHP9 54587248 IC50 > 10000 nM T59654 CE1ZK6 54759168 IC50 > 10000 nM T59654 C6QGO9 56657855 IC50 > 10000 nM T59654 CBZ8T4 56657856 IC50 = 335 nM T59654 CA6T5S 56664839 IC50 > 10000 nM T59654 CYZ57N 56668250 IC50 > 10000 nM T59654 CYPL60 56675140 IC50 > 10000 nM T59654 CTBX87 56681780 IC50 > 10000 nM T59654 CH53XJ 57391650 IC50 > 10000 nM T59654 CF4U0R 57391651 IC50 > 10000 nM T59654 CRLG52 57395119 IC50 > 10000 nM T59654 CX6GJ7 57396885 IC50 > 10000 nM T59654 CG4D3H 57398639 IC50 > 10000 nM T59654 CMQ7A6 57400314 IC50 > 10000 nM T59654 CEG5Q7 57403865 IC50 > 10000 nM T59654 CK7L8O 57403866 IC50 > 10000 nM T59654 CTV3K8 58405292 IC50 = 25 nM T59654 CNM93S 58405323 IC50 = 9 nM T59654 CCZ98N 58405467 IC50 = 2990 nM T59654 CC90XE 58405504 IC50 = 130 nM T59654 C29QLR 58405566 IC50 = 1150 nM T59654 C8RGV3 58405571 IC50 = 15 nM T59654 CE69UL 58405593 IC50 = 31 nM T59654 C2O3YU 58405631 IC50 = 5 nM T59654 C2L5SP 58405634 IC50 = 168 nM T59654 C8QE2P 58405636 IC50 = 60 nM T59654 CE38BL 58405673 IC50 = 1870 nM T59654 CJG5F1 58405732 IC50 = 740 nM T59654 CC8OS6 58405741 IC50 = 1040 nM T59654 CL7TF1 58405755 IC50 = 2710 nM T59654 CYN56J 58405790 IC50 = 354.7 nM T59654 CDNU35 58405817 IC50 = 2560 nM T59654 C41DJO 58405910 IC50 = 12 nM T59654 CDGV17 58405948 IC50 = 5820 nM T59654 CG63RM 58415665 IC50 = 30 nM T59654 CV63UL 67240318 IC50 = 310 nM T59654 CKT60L 71455860 Ki = 2 nM T59654 C05ICM 71602777 IC50 = 13 nM T59654 CD7U3Q 71602778 IC50 = 8 nM T59654 C7BVZ4 71602779 IC50 = 21 nM T59654 CGOI91 71602780 IC50 = 2050 nM T59654 C64YHA 71602828 IC50 = 17 nM T59654 C9B7LV 71602829 IC50 = 44 nM T59654 CDSP70 71602874 IC50 = 532 nM T59654 CUF0G5 71602875 IC50 = 120 nM T59654 CP0OI3 73353560 IC50 = 3870 nM T59654 C7E2JD 73353563 IC50 = 3190 nM T59654 C0Q1FT 91938009 IC50 > 50000 nM T59654 CGB54P 101902999 IC50 = 10000 nM T59654 C34EVY 134143682 IC50 = 290 nM T59654 C0CM9H 135879715 IC50 = 8900 nM T59654 C01HMT 135932346 IC50 > 10000 nM T59654 C4RL7Q 135985508 IC50 > 10000 nM T59654 C8WIM5 135985510 IC50 > 10000 nM T59654 C3M7EP 135985511 IC50 = 5700 nM T59654 CMQ5W9 135985512 IC50 > 10000 nM T59654 CGM2H4 135988906 IC50 > 10000 nM T59654 CXM18S 135988925 IC50 > 10000 nM T59654 C1ZT4N 135988927 IC50 > 10000 nM T59654 CVG5B9 135988940 IC50 = 4400 nM T59654 C68JXP 135988944 IC50 > 10000 nM T59654 CG23XF 135988947 IC50 > 10000 nM T59654 CIFX04 135988950 IC50 > 10000 nM T59654 CGP53C 135988956 IC50 > 10000 nM T59654 CLNJ17 135988957 IC50 > 10000 nM T59654 C7NU6A 135988961 IC50 > 10000 nM T59654 CR81AC 135988980 IC50 > 10000 nM T59654 C86BZJ 135988997 IC50 > 10000 nM T59654 C80PXZ 135989011 IC50 = 10000 nM T59654 CC6SO7 135989013 IC50 > 10000 nM T59654 CY57SZ 136239319 IC50 < 10000 nM T59654 CJ2L3P 136239450 IC50 = 1900 nM T59654 C7XY0Q 136239451 IC50 > 10000 nM T59654 CN5LQ2 136239452 IC50 = 10000 nM T59654 CY08AS 136244133 IC50 > 10000 nM T59654 CH8YL3 137632392 IC50 = 250 nM T59654 C0XP4L 137632541 IC50 = 3400 nM T59654 C0UE7N 137648535 IC50 = 3500 nM T59654 CN1LP0 137652774 IC50 = 310 nM T59654 CNP59S 141451364 IC50 = 8.16 nM T59654 C7QXC6 141451369 IC50 = 4.72 nM T59654 CM7O6D 141451370 IC50 = 265.1 nM T59654 CYHN75 141451372 IC50 = 3.4 nM T59654 CK1I8G 141451381 IC50 = 23.87 nM T59654 C6KQ8V 141451382 IC50 = 19.85 nM T59654 CRIZ46 141451383 IC50 = 498 nM T59654 C0QO5H 141451384 IC50 = 626.2 nM T59654 C78KWO 141451386 IC50 = 54.4 nM T59654 C09NZC 141451387 IC50 = 36.04 nM T59654 CJ21FB 145949301 IC50 = 478.3 nM T59654 CA0RG8 145949395 IC50 = 124.5 nM T59654 CCS05D 145950319 IC50 = 384.3 nM T59654 C6LBJ2 145950482 IC50 = 18.62 nM T59654 C5L2IY 145950845 IC50 = 158.8 nM T59654 CDT45G 145951146 IC50 = 4.88 nM T59654 CJ0H6I 145951269 IC50 = 17.41 nM T59654 C6J2FE 145951598 IC50 = 71.55 nM T59654 CWP5K3 145952451 IC50 = 969.2 nM T59654 CAD7R9 145953240 IC50 = 242.5 nM T59654 CEKL79 145954798 IC50 = 1500 nM T59654 CH0FJ8 145955296 IC50 = 189.6 nM T59654 CJ96ZH 145955626 IC50 = 311 nM T59654 C3TQ1E 145955731 IC50 = 10.17 nM T59654 C1AYV7 145957415 IC50 = 16.52 nM T59654 C5J7AZ 145957656 IC50 = 159 nM T59654 C39VOT 145958071 IC50 = 217.7 nM T59654 C9NPH7 145958192 IC50 = 28.51 nM T59654 CFGI54 145958286 IC50 = 8.6 nM T59654 C98TDA 145958548 IC50 = 90.93 nM T59654 C1BJS3 145958954 IC50 = 120.6 nM T59654 C5KRP1 145960780 IC50 = 11.35 nM T59654 CD3K7O 145961079 IC50 = 13370 nM T59654 CKJN89 145961654 IC50 = 21.77 nM T59654 CL56JT 145963032 IC50 = 715.7 nM T59654 C63ELA 145963541 IC50 = 206.7 nM T59654 CQP70K 145971255 IC50 = 7.86 nM T59654 CV4G1E 145973188 IC50 = 17.77 nM T59654 C7JIR5 145973809 IC50 = 7.06 nM T59654 CVU71O 145975475 IC50 = 192 nM T59654 C64XYG 145975479 IC50 = 190.7 nM T59654 C1MA9Q 145979724 IC50 = 150 nM T59654 C90QCO 145980261 IC50 = 110 nM T59654 CSY3K4 145987182 IC50 = 610 nM T59654 CY18PZ 145990069 IC50 = 3100 nM T59654 C2MD1Q 155513187 IC50 > 10000 nM T59654 CQA75Z 155514946 IC50 = 61.17 nM T59654 CH82NV 155516034 IC50 = 718.3 nM T59654 CQST37 155519017 IC50 = 167.3 nM T59654 CEI34U 155519091 IC50 = 131.7 nM T59654 CV40JF 155519344 IC50 = 85.11 nM T59654 C67ARO 155520726 IC50 > 10000 nM T59654 C1SWX6 155520963 IC50 = 75.77 nM T59654 CUSF64 155521348 IC50 = 338.7 nM T59654 CTZ07V 155523554 IC50 = 1796.9 nM T59654 CB2LE0 155524979 IC50 = 107.2 nM T59654 C0P5XN 155525853 IC50 = 33.83 nM T59654 C4D3WX 155526889 IC50 = 30.51 nM T59654 CM1HB6 155527327 IC50 = 122.2 nM T59654 C9JT8G 155528462 IC50 = 290.5 nM T59654 C73EUH 155530844 IC50 = 643 nM T59654 CD65ZS 155533233 IC50 = 3474 nM T59654 CCL97M 155533912 IC50 > 10000 nM T59654 CUI36R 155536170 IC50 > 10000 nM T59654 CRWI29 155538752 IC50 > 10000 nM T59654 CM71YQ 155539415 IC50 = 743.9 nM T59654 CA9H6Y 155539913 IC50 = 3180 nM T59654 CKR8W0 155541766 IC50 = 230.9 nM T59654 C69LPE 155543442 IC50 = 195.9 nM T59654 CMR1S9 155545273 IC50 = 385.3 nM T59654 CC1MU2 155546554 IC50 = 152 nM T59654 CB9V4S 155549112 IC50 = 7.98 nM T59654 C7R1IQ 155551215 IC50 = 868.7 nM T59654 CN5D6K 155552906 IC50 = 314.2 nM T59654 C6C1DL 155553924 IC50 = 873.6 nM T59654 CSDM31 155562825 IC50 = 107 nM T59654 CU9HL1 155563487 IC50 = 397.3 nM T59654 C21DOA 155564098 IC50 = 640.8 nM T59654 CC1MR2 155566593 IC50 = 898.4 nM T59654 C3XS1Q 155568979 IC50 = 3.98 nM T59654 D0W7TU 947057 IC50 > 50000 nM T64591 D00XWD 135409453 Ki = 2511.89 nM T64591 D01AZG 5073 Ki > 1000 nM T64591 D03WEX 9966051 Ki = 3.7 nM T64591 D04FVU 6337614 Ki = 0.03162 nM T64591 D04QSJ 3052762 Ki = 3981.07 nM T64591 D05ZIK 4205 Ki = 2900 nM T64591 D06GKN 2099 Ki = 0.5 nM T64591 D0G8NN 119570 Ki > 10000 nM T64591 D0H3HM 60795 Ki = 1000 nM T64591 D0H7KF 5002 Ki > 1000 nM T64591 D0K0KH 656665 Ki = 2.7 nM T64591 D0K7WK 4595 IC50 = 0.09 nM T64591 D0RA9E 108000 Ki = 0.06 nM T64591 D0U2OO 2477 Ki > 10000 nM T64591 D0V4QS 135398745 Ki = 1000 nM T64591 D0Z1RV 135398737 Ki = 186.21 nM T64591 D0Z6UC 5358 IC50 = 9.3 nM T64591 D01HVZ 11961293 Ki = 100000 nM T64591 D05LRD 59286554 IC50 = 8100 nM T64591 D06QZL 65997 Ki = 0.36 nM T64591 D0D3TX 46196517 IC50 = 299 nM T64591 D0L3JI 188942 Ki = 750 nM T64591 D0LI1C 44469321 IC50 > 10000 nM T64591 D0N5KS 154104 EC50 = 5.4 nM T64591 D0R2OU 25070031 Ki = 2 nM T64591 D0W5EH 6918388 IC50 < 6 nM T64591 D0X2XF 177336 Ki > 1000 nM T64591 D02ZSO 6426760 IC50 > 10000 nM T64591 D0K1SZ 3019427 EC50 = 2300 nM T64591 D0L9YS 4581 EC50 = 24 nM T64591 D0Q9RR 9794392 Ki = 12 nM T64591 D0V3GT 671690 Ki = 2.5 nM T64591 D0ZG9N 132337 Ki = 152 nM T64591 CZUI83 2769 Ki = 1995.26 nM T64591 C5H9CN 9287 Ki > 10000 nM T64591 CIMO04 11385 Ki = 1000 nM T64591 CTB26S 52899 Ki > 10000 nM T64591 CAF7T8 64622 Ki > 1000 nM T64591 CX1GC4 108182 Ki = 0.39 nM T64591 CKP25M 121881 Ki = 158.49 nM T64591 CFBY39 129150 Ki = 794.33 nM T64591 CF1O8E 130946 Ki = 1 nM T64591 CVZW19 182593 Ki = 1995.26 nM T64591 CX30KB 720937 IC50 = 620 nM T64591 CZN6S9 743974 EC50 > 50118.72 nM T64591 C2VLP8 752521 Ki > 10000 nM T64591 C0RIJ7 1403136 Ki = 0.05129 nM T64591 CQL9G3 2737193 Ki = 19.21 nM T64591 C3C6AI 3035572 Ki = 0.42 nM T64591 C32RYW 3044599 Ki = 537.03 nM T64591 CAM8H3 3066250 IC50 > 1000 nM T64591 CR1PZ2 3513127 Ki = 794.33 nM T64591 CS8KE2 3649661 Ki > 10000 nM T64591 CUBH90 6604794 Ki = 0.1445 nM T64591 CY1XN7 7446712 IC50 = 1000 nM T64591 C6HQB2 9793921 Ki = 1258.93 nM T64591 C6YDQ0 9795278 Ki = 930 nM T64591 CK0U5Q 9797360 IC50 > 3160 nM T64591 CR8ET5 9814387 Ki = 56 nM T64591 CC24WR 9845261 IC50 > 100000 nM T64591 CM13ZV 9856041 Ki > 10000 nM T64591 C0ZR3E 9861687 IC50 > 1000 nM T64591 C5WYN4 9865858 Ki > 1000 nM T64591 CB7J1X 9879256 IC50 > 3160 nM T64591 CBF9T3 9879532 Ki = 36 nM T64591 C9J6KN 9901423 Ki = 190 nM T64591 CYWQ50 9906447 Ki > 10000 nM T64591 CWJ0I1 9906933 Ki = 1 nM T64591 COD73F 9943346 IC50 = 580 nM T64591 C2RU8Q 9966169 Ki = 440 nM T64591 CR84AX 9970357 Ki = 2 nM T64591 C9XUH5 9976826 Ki = 60 nM T64591 C1XK9Y 10019102 IC50 > 10000 nM T64591 C2EUY0 10035109 Ki > 10000 nM T64591 C2C1XS 10042602 Ki < 10000 nM T64591 C6VO4P 10046170 Ki > 1000 nM T64591 CQVJ58 10088453 Ki < 10000 nM T64591 CJK86Q 10192961 IC50 = 150 nM T64591 CG2B7I 10247701 Ki = 5248.07 nM T64591 CMNH04 10286136 IC50 = 484 nM T64591 CA3E4W 10316297 Ki > 10000 nM T64591 C74KUP 10336265 Ki = 0.42 nM T64591 CN8PA7 10357986 IC50 > 10000 nM T64591 CNJ03F 10374840 Ki = 32 nM T64591 C69KIB 10385855 IC50 > 10000 nM T64591 C3RPH6 10425296 Ki = 1 nM T64591 CLDM93 10445840 Ki = 310 nM T64591 C48BRW 10546334 Ki = 5248.07 nM T64591 CU45KX 10656971 Ki = 4.677 nM T64591 C4SBO9 10915140 IC50 > 10000 nM T64591 CHLQ20 11004759 Ki = 0.33 nM T64591 C2CB4G 11174673 Ki = 26 nM T64591 CL49OC 11178730 IC50 > 100 nM T64591 C8WHY7 11190823 IC50 = 48.4 nM T64591 C7Q4LE 11213399 IC50 = 26.7 nM T64591 C20HPU 11220991 IC50 = 779 nM T64591 CWF6A1 11305391 IC50 = 99.4 nM T64591 CA0F6Z 11311114 Ki = 579 nM T64591 CP4K5G 11328306 IC50 = 84.8 nM T64591 CBO7W4 11329644 IC50 = 100 nM T64591 C4DV2B 11339853 IC50 = 46.5 nM T64591 CU6CR4 11374124 IC50 = 45.6 nM T64591 CQU73N 11376655 Ki = 5.6 nM T64591 C85LYP 11430418 Ki = 4.72 nM T64591 CN6F9K 11464531 IC50 = 45.7 nM T64591 COMY40 11476372 IC50 = 48.3 nM T64591 C9ZT5F 11536299 Ki = 2511.89 nM T64591 CYG3H9 11543786 Ki = 174 nM T64591 C18BAJ 11572597 IC50 = 3310 nM T64591 C83DCU 11609760 IC50 > 7310 nM T64591 CN4Z5C 11679149 IC50 = 19952.62 nM T64591 C3M8DW 11709098 IC50 = 70 nM T64591 CZ2EX9 11724799 Ki = 53.2 nM T64591 CBNC94 11752512 IC50 = 41.4 nM T64591 C8JQL7 11957735 IC50 > 10000 nM T64591 CTXK62 12686479 Ki = 12.59 nM T64591 CP6ZT4 12706835 Ki = 407.38 nM T64591 CRJ4X2 12741697 Ki = 251.19 nM T64591 C8ZAJ9 13025568 Ki = 1.622 nM T64591 CHK8W2 14722779 Ki = 1 nM T64591 C4F1UJ 14742526 Ki = 12 nM T64591 CYW76P 14742527 Ki = 1.8 nM T64591 CZ70OA 14742528 Ki = 1.94 nM T64591 C7X4LQ 15046233 Ki = 64 nM T64591 C4O0LJ 15636963 Ki = 3.3 nM T64591 CZ2IS9 16660294 Ki > 10000 nM T64591 COJU37 16727124 Ki = 47.3 nM T64591 C3W8ZK 17758335 IC50 = 30000 nM T64591 COF61U 17982621 Ki = 49.8 nM T64591 COWC18 19786480 Ki = 5.21 nM T64591 C3T5HF 21509921 Ki > 10000 nM T64591 CQB20R 23155620 IC50 > 100 nM T64591 CZ25WJ 23155621 IC50 > 100 nM T64591 CM57CZ 23155625 IC50 = 63.8 nM T64591 CFB0G1 23155644 IC50 > 100 nM T64591 C7FQU2 23155650 IC50 = 59.1 nM T64591 C8Y7LC 23155667 IC50 = 15.6 nM T64591 C1PX5S 23155676 IC50 > 100 nM T64591 CC46FD 23155688 IC50 > 100 nM T64591 CAC0S3 23155689 IC50 = 50.5 nM T64591 C57WEZ 23155758 IC50 = 83.1 nM T64591 CXHB39 23155770 IC50 = 97.9 nM T64591 C1OVU4 23155818 IC50 > 100 nM T64591 CKQ2Y0 23155825 IC50 > 100 nM T64591 C2NOU7 23155834 IC50 = 62.1 nM T64591 C75GWQ 23155840 IC50 > 100 nM T64591 C1N6SD 23155860 IC50 = 69.9 nM T64591 CTC8Y5 23155869 IC50 > 100 nM T64591 CK3PM5 23155885 IC50 > 100 nM T64591 C8XYR2 23155900 IC50 > 100 nM T64591 CFG6D5 23155906 IC50 > 100 nM T64591 CQS93U 23155935 IC50 > 100 nM T64591 C3P1TG 23155946 IC50 = 87.6 nM T64591 C5LCT7 23155948 IC50 = 64.8 nM T64591 C6QCL8 23155950 IC50 > 100 nM T64591 C7DQ5C 23155951 IC50 = 61 nM T64591 C7PSB8 23155955 IC50 > 100 nM T64591 CXR3G9 23155963 IC50 > 100 nM T64591 CC1P4X 23155976 IC50 = 44.2 nM T64591 CJY62P 23155980 IC50 > 100 nM T64591 CXWI74 23332842 IC50 = 19000 nM T64591 CV4GM7 24178523 Ki = 0.6 nM T64591 CO01RG 24178536 Ki = 32.7 nM T64591 CTZL46 24278976 Ki = 0.04 nM T64591 CAVZ24 24759518 Ki = 12.02 nM T64591 CQ5S2G 24759622 Ki = 1.349 nM T64591 C6P4SW 24769782 Ki = 12.9 nM T64591 CVR27S 24769783 Ki = 2.4 nM T64591 CE2XP4 24795080 Ki = 700 nM T64591 C09OLY 24804735 IC50 = 1900 nM T64591 CY21RE 24841480 Ki = 1900 nM T64591 CIR64L 24860582 IC50 > 30000 nM T64591 C5YRN3 24995682 Ki = 2 nM T64591 C69KXY 24995990 Ki = 8.9 nM T64591 CF2AH1 24995991 Ki = 1.6 nM T64591 CB5LR3 24995992 Ki = 7.9 nM T64591 CEW1L6 24995993 Ki = 4.8 nM T64591 C3N5HP 24995994 Ki = 1.9 nM T64591 C3F8BL 24995995 Ki = 13 nM T64591 CSX8R9 24995996 Ki = 8.1 nM T64591 CJM8R0 24996322 EC50 = 1.1 nM T64591 CE31GM 24996323 Ki = 7.8 nM T64591 C5N6PJ 24996324 Ki = 5.3 nM T64591 CPL5O0 24996325 Ki = 1.8 nM T64591 CF7R8J 24996326 Ki = 2.5 nM T64591 CED80Q 24996327 Ki = 1.7 nM T64591 C12YIC 24996643 Ki = 3 nM T64591 CL0RC1 24996649 Ki = 11 nM T64591 CXRZ70 24997749 IC50 > 30000 nM T64591 CHD36Z 24998360 IC50 > 30000 nM T64591 C5V1YO 25029711 IC50 > 31622.78 nM T64591 CBY3O2 25070582 IC50 = 2300 nM T64591 CAGM54 25129523 Ki = 1258.93 nM T64591 CQR84M 25147644 Ki > 10000 nM T64591 C6HD3B 25147771 Ki = 2.818 nM T64591 C0AG1S 25178131 Ki = 79.43 nM T64591 CXWJ98 25178132 Ki = 165.96 nM T64591 C9R3VG 25178339 Ki = 16595.87 nM T64591 CXF28Y 25178341 Ki = 2.692 nM T64591 CLVH57 25178344 Ki = 14.79 nM T64591 C5FMI4 25178558 Ki = 3548.13 nM T64591 CJ5EH8 25178933 Ki = 13.8 nM T64591 C7C9LH 25178936 Ki = 6.607 nM T64591 C59YLX 25178937 Ki = 1.122 nM T64591 C2Y3JU 25179300 Ki = 18.2 nM T64591 CX38LG 25179302 Ki = 2344.23 nM T64591 CYW92S 25179305 Ki = 11748.98 nM T64591 CS63PT 25191018 IC50 = 800 nM T64591 CR3F9D 25196518 IC50 = 1600 nM T64591 CWGM20 25196628 IC50 = 2100 nM T64591 C9IR0F 25196631 IC50 = 1400 nM T64591 C3RLZ5 25196632 IC50 = 2700 nM T64591 CWTO86 25196740 IC50 = 2200 nM T64591 CI29CP 25196741 IC50 = 2200 nM T64591 C0X1TL 25196744 IC50 = 2800 nM T64591 CPAR05 25196745 IC50 = 1300 nM T64591 CA58DL 41305446 Ki > 10000 nM T64591 C1CWU0 42631007 IC50 = 251188.64 nM T64591 CJ3NP5 42636941 IC50 = 6.918 nM T64591 CK7F2E 44240743 IC50 > 30000 nM T64591 C4W0SH 44247585 IC50 = 480 nM T64591 CD2E1H 44307643 Ki = 1.69 nM T64591 CJ6QD5 44307771 EC50 = 240 nM T64591 CQ23ET 44307976 Ki = 7.96 nM T64591 CG5QZ6 44307990 Ki = 1.43 nM T64591 CHX45P 44307991 Ki = 7.43 nM T64591 CAS3C2 44362829 Ki = 0.138 nM T64591 CG9Y5H 44408892 Ki > 100000 nM T64591 COX8D7 44408895 Ki > 100000 nM T64591 CR6CE1 44408940 Ki > 100000 nM T64591 C3HCS5 44419820 IC50 = 275 nM T64591 CWTD76 44422208 IC50 = 57000 nM T64591 CM8YH1 44422216 IC50 = 2100 nM T64591 CB26HU 44422228 IC50 = 19800 nM T64591 CWM49B 44422255 IC50 = 15800 nM T64591 CGRF72 44422338 IC50 = 5900 nM T64591 CYG93V 44427853 Ki = 3100 nM T64591 C3C2OK 44427854 Ki = 10000 nM T64591 C8Y9FW 44427856 Ki = 19000 nM T64591 C19LSU 44427858 Ki = 100000 nM T64591 C1FY4M 44427860 Ki = 15000 nM T64591 CC2BE1 44427862 Ki > 100000 nM T64591 CW95BM 44427864 Ki = 2511.89 nM T64591 C3XJ4Z 44427866 Ki = 100000 nM T64591 C84GXL 44427868 Ki = 25118.86 nM T64591 C8CPX2 44427870 Ki = 5700 nM T64591 CS17TJ 44427872 Ki = 23000 nM T64591 CDL67C 44427876 Ki = 1900 nM T64591 C9B6ER 44427877 IC50 = 3981.07 nM T64591 C15UHM 44427879 IC50 = 30000 nM T64591 CCAV10 44427881 IC50 = 30000 nM T64591 CXRV71 44427883 IC50 = 30000 nM T64591 CKX81C 44427885 Ki > 100000 nM T64591 CZL97F 44455426 Ki > 10000 nM T64591 C6BFI0 44456033 Ki = 1062.3 nM T64591 C12XGE 44456400 Ki = 34 nM T64591 C4DL5C 44469677 IC50 > 10000 nM T64591 C6WV2P 44559406 IC50 > 100000 nM T64591 CVA67X 44568347 Ki = 3900 nM T64591 C5TKU6 44579715 Ki = 3260 nM T64591 CRCH48 44582675 Ki > 10000 nM T64591 CEJ4R8 44582676 Ki > 10000 nM T64591 CZGP86 44582677 Ki > 10000 nM T64591 C5QB4K 44582678 Ki > 10000 nM T64591 C01RCI 44582705 Ki > 10000 nM T64591 CXL25V 44582706 Ki > 10000 nM T64591 C8MR1X 44582707 Ki > 10000 nM T64591 C4IT1N 44582708 Ki > 10000 nM T64591 CB0S4Z 44592109 IC50 > 10000 nM T64591 CC52XI 44592242 Ki > 10000 nM T64591 CFSB52 44592414 Ki = 251.19 nM T64591 C7TD8N 44611609 IC50 > 30000 nM T64591 C0ZF2L 44611611 IC50 > 30000 nM T64591 C5Q2CN 44611748 IC50 > 30000 nM T64591 CS9GW5 44611875 IC50 > 30000 nM T64591 CO3I5F 44622849 Ki = 3700 nM T64591 CNR3K1 44626294 IC50 = 18 nM T64591 C5ABG6 44626295 IC50 = 159 nM T64591 CXYK56 45268365 Ki = 3993 nM T64591 CT0Y4W 45485562 IC50 = 4900 nM T64591 CE9D2C 45485563 IC50 = 3500 nM T64591 CSML06 45485564 IC50 = 1400 nM T64591 CQU3S9 45485604 IC50 = 1600 nM T64591 CG5QJ0 45485614 IC50 = 3100 nM T64591 CE4ZG1 45485619 IC50 = 2500 nM T64591 CSK1X6 45485620 IC50 = 790 nM T64591 CCY98N 45485624 IC50 = 390 nM T64591 CREQ49 45485653 IC50 = 1700 nM T64591 CTQ1U3 45485675 IC50 = 2800 nM T64591 CR0I3A 46180744 IC50 = 2480 nM T64591 CKI1P8 46233560 Ki = 26.3 nM T64591 CHCR01 46233590 Ki = 375 nM T64591 CP5EJ2 46233591 Ki = 7.3 nM T64591 C4VX8P 46233592 Ki = 5306 nM T64591 C3BIO6 46233593 Ki = 3029 nM T64591 C3WG4A 46233633 Ki = 237 nM T64591 C85NEI 46233634 Ki = 749 nM T64591 C75HQN 46233635 Ki = 0.67 nM T64591 C0VJ8U 46233636 Ki = 71.1 nM T64591 CSVZ12 46233637 Ki = 0.23 nM T64591 CNCD06 46233671 Ki = 59.3 nM T64591 CKE13P 46831056 IC50 = 7800 nM T64591 CFUP50 46831057 IC50 = 5700 nM T64591 C4DVF7 46831058 IC50 = 5800 nM T64591 CXOC17 46831059 IC50 > 30000 nM T64591 CL98UY 46831060 IC50 > 30000 nM T64591 CBR46Y 46831061 IC50 > 30000 nM T64591 C03LTM 46869265 Ki = 870000 nM T64591 C7JB8W 46906000 IC50 = 2800 nM T64591 C2LZJ0 49783209 Ki = 1072 nM T64591 C57SMG 49783415 Ki = 3511 nM T64591 C0TG6I 49783419 Ki > 10000 nM T64591 COE79D 49836152 IC50 > 100 nM T64591 C6IN7B 49836154 IC50 = 86.6 nM T64591 C8JQ4O 49837354 IC50 = 77.6 nM T64591 CN0MO8 49837461 IC50 = 50.6 nM T64591 CHB1I9 49837652 IC50 = 22.1 nM T64591 CG64FA 49837758 IC50 = 52.6 nM T64591 CY46CB 49843532 Ki = 8.1 nM T64591 CC1SF7 49863118 IC50 = 7943.28 nM T64591 C2RY0J 50878551 Ki > 10000 nM T64591 C1W6TV 50898777 Ki = 2511.89 nM T64591 CXMZ73 50898778 Ki > 10000 nM T64591 CX48AD 51002362 IC50 > 10000 nM T64591 CE4KP1 51050257 Ki > 10000 nM T64591 CK8J4G 52108285 Ki = 2.951 nM T64591 CL2P8X 52920232 IC50 = 12000 nM T64591 C42ROG 52920234 IC50 = 350 nM T64591 CCP0V7 52920236 IC50 = 9200 nM T64591 C6XW8S 52940690 Ki = 36.4 nM T64591 CM4XO6 52941718 Ki > 1000 nM T64591 CDV52R 52941871 Ki = 66.5 nM T64591 C0F3LG 52943305 Ki = 165 nM T64591 C34ZMB 52945520 Ki = 13.8 nM T64591 C3CGW6 52946744 Ki = 18.2 nM T64591 CLG7C6 52947945 Ki = 6.8 nM T64591 CZ84TY 52949185 Ki = 36.4 nM T64591 CX2MZ4 52949186 Ki = 12.4 nM T64591 CN85WP 52949210 Ki = 4.7 nM T64591 C4MZ1V 53237227 Ki = 310 nM T64591 CBIL92 53237431 Ki = 500 nM T64591 C7L6PJ 53237434 Ki = 260 nM T64591 C9UX5B 53237437 Ki = 36 nM T64591 CMV78H 53237440 Ki = 53 nM T64591 CL73GJ 53237662 Ki = 140 nM T64591 CS02ZU 53237664 Ki = 450 nM T64591 C5MLV8 53237666 Ki = 62 nM T64591 CLUD12 53237668 Ki = 64 nM T64591 C9P7KL 53237670 Ki = 52 nM T64591 C8T9OE 53237672 Ki = 32 nM T64591 COJM04 53237674 Ki = 86 nM T64591 C4TNP6 53237891 Ki = 110 nM T64591 C9RIJ7 53237893 Ki = 33 nM T64591 CBZX08 53237895 Ki = 80 nM T64591 C5ZT7N 53237897 Ki = 67 nM T64591 C4KRV8 53237899 Ki = 29 nM T64591 CNJ02E 53237901 Ki = 32 nM T64591 C0H6TR 53237903 Ki = 26 nM T64591 C8TDE6 53238121 Ki = 12 nM T64591 CN4R7I 53238123 Ki = 17 nM T64591 CIP64Q 53238125 Ki = 7.3 nM T64591 C70LGK 53238127 Ki = 160 nM T64591 C2WK6F 53238129 Ki = 150 nM T64591 C6C0KM 53238131 Ki = 45 nM T64591 CXN12U 53238133 Ki = 670 nM T64591 C9QXC8 53238134 Ki = 130 nM T64591 C9Z3FA 53238355 Ki = 27 nM T64591 C1Z8AH 53238357 Ki = 270 nM T64591 CMJ62D 53245590 Ki = 1000 nM T64591 C3Y4WN 53316626 Ki = 0.7 nM T64591 CB03KI 53323199 Ki = 0.9 nM T64591 CU59EZ 53363442 Ki = 2.8 nM T64591 C8WHT5 56593934 Ki = 10000 nM T64591 C53IST 56672434 Ki = 1.585 nM T64591 CBW5E1 56946195 Ki = 19 nM T64591 C4P7LC 56946196 Ki = 2.7 nM T64591 C1TC7Q 56963799 Ki > 10000 nM T64591 C2PW6U 57486204 IC50 = 11000 nM T64591 CHI0M1 57486210 IC50 = 2300 nM T64591 C31TNG 57523356 IC50 > 30000 nM T64591 CEV26F 57523382 IC50 > 30000 nM T64591 CHK96S 57523383 IC50 > 30000 nM T64591 CKV91C 57523414 IC50 > 30000 nM T64591 CK76WH 57523415 IC50 > 30000 nM T64591 C2E4CS 57523447 IC50 > 30000 nM T64591 C9IU7S 58081849 IC50 = 71000 nM T64591 COT69D 58081856 IC50 = 1700 nM T64591 CE8V0W 58081870 IC50 = 44000 nM T64591 C2UZ1H 58087975 IC50 = 21 nM T64591 CG2DS4 58087977 IC50 = 14000 nM T64591 C7O3GZ 58088026 IC50 = 54 nM T64591 C9V8HI 58088056 IC50 = 23 nM T64591 CEV8F6 58088113 IC50 = 16 nM T64591 CND4G1 58088117 IC50 = 34000 nM T64591 CMY5N3 58088118 IC50 = 15 nM T64591 CO14JV 58088126 IC50 = 3800 nM T64591 C9CJO2 58088140 IC50 = 20000 nM T64591 C2XEH4 58088161 IC50 = 19000 nM T64591 C7ZBE4 58088162 IC50 = 25 nM T64591 CC18WB 58088207 IC50 = 8100 nM T64591 CKW02I 59173799 IC50 > 31622.78 nM T64591 CH6ZY0 59286581 IC50 = 85 nM T64591 CUNG95 60132884 Ki = 12 nM T64591 CXKD25 66810955 Ki = 100000 nM T64591 C40FKD 66898172 Ki = 13.5 nM T64591 C7TJ9X 66898814 Ki = 6.4 nM T64591 C1LEH8 67268994 Ki > 10000 nM T64591 CWH4A1 69604399 Ki = 1.445 nM T64591 CN1T4U 69925573 IC50 = 180 nM T64591 C9N3VB 69937087 Ki = 0.2 nM T64591 CHD80I 69937162 Ki = 0.5 nM T64591 CAR2N8 69937236 Ki = 3.1 nM T64591 CN7X0U 69937257 Ki = 5.7 nM T64591 CD86LU 69937258 Ki = 67.6 nM T64591 CY7G9I 69937654 Ki = 701 nM T64591 C6ICU8 70896220 Ki = 0.8 nM T64591 C3XNC2 71450247 Ki = 2470 nM T64591 C9GDI4 71451613 Ki = 13.49 nM T64591 CW8G1Z 71453451 Ki = 5.888 nM T64591 CE7U4Q 71453797 Ki = 18600 nM T64591 CAQF34 71455625 Ki = 641 nM T64591 CDL61M 71456956 Ki = 331.13 nM T64591 C7MNB5 71457264 IC50 > 10000 nM T64591 CMJ1O9 71457409 Ki > 10000 nM T64591 C3RC2E 71458823 Ki = 204.17 nM T64591 CS83IF 71459269 Ki = 410 nM T64591 CP5MZ1 71460633 Ki = 467.74 nM T64591 C5OV1C 71460637 Ki = 7.413 nM T64591 C63YLA 71461049 Ki > 10000 nM T64591 CJD96I 71461050 Ki = 710 nM T64591 C8S3NJ 71462343 Ki = 218.78 nM T64591 C4P3JU 71462776 Ki = 1314 nM T64591 C3GUQ2 71462777 Ki = 680 nM T64591 CL91AC 71463022 Ki = 7612 nM T64591 CUG93T 71712325 Ki = 15848.93 nM T64591 CZ0C2S 71712326 Ki = 1258.93 nM T64591 CJF19S 71712327 Ki = 100000 nM T64591 C2HBK3 71712328 Ki = 79432.82 nM T64591 CUG29A 71712329 Ki = 39810.72 nM T64591 CZ5B9H 71712463 Ki = 79432.82 nM T64591 CT2I5Z 71712464 Ki = 50118.72 nM T64591 C4EXG5 71712465 Ki = 63095.73 nM T64591 C98QJG 71712466 Ki = 100000 nM T64591 C0RDS6 71712611 Ki = 50118.72 nM T64591 C9J8ST 71712612 Ki = 19952.62 nM T64591 CL6RN0 71712613 Ki = 63095.73 nM T64591 CIH6T3 71714540 Ki = 79432.82 nM T64591 CJ2SI1 71714541 Ki = 79432.82 nM T64591 CJQ45N 71714542 Ki = 50118.72 nM T64591 C8RO7X 71714543 Ki = 39810.72 nM T64591 CS0YC8 71714544 Ki = 7943.28 nM T64591 CINY69 72192461 IC50 = 7400 nM T64591 CWH6T3 72548703 IC50 = 4.9 nM T64591 C8Z0NM 72550642 Ki > 10000 nM T64591 CL6W2Q 72550645 Ki > 10000 nM T64591 C78LYM 72698087 Ki = 1200 nM T64591 C63HPK 72698088 Ki = 2600 nM T64591 C6NOM3 72703256 Ki = 230 nM T64591 C0GQ7F 72703471 Ki = 505 nM T64591 CSW89Y 72709023 IC50 = 32000 nM T64591 CQ30RG 72709025 IC50 > 12000 nM T64591 C9AD0M 72709102 IC50 = 5600 nM T64591 C0JXT9 72709105 IC50 = 26 nM T64591 C6QOL9 72709106 IC50 = 43 nM T64591 C12AOM 72709107 IC50 = 860 nM T64591 C48SNQ 72709187 IC50 = 620 nM T64591 CA2BX4 72709190 IC50 > 100000 nM T64591 CA94ZJ 72709267 IC50 = 14500 nM T64591 CXA2P7 72709272 IC50 = 32000 nM T64591 CNGR78 72709273 IC50 = 13000 nM T64591 CH2RT8 72709349 IC50 = 1400 nM T64591 C1K9OD 72709587 IC50 = 18000 nM T64591 COH37Y 72709588 IC50 = 38 nM T64591 CZB6J7 72709589 IC50 = 51 nM T64591 CLM6P9 72709673 IC50 = 26 nM T64591 CL01VG 72709675 IC50 = 6400 nM T64591 CCM45B 72709679 IC50 = 38000 nM T64591 CSDO19 72709764 IC50 = 47000 nM T64591 CP52FZ 72709766 IC50 = 170 nM T64591 CF8W5S 72709767 IC50 = 64000 nM T64591 C56HYB 72710014 IC50 = 61000 nM T64591 CC6Q5R 72771081 Ki < 100 nM T64591 CC65OA 73213195 Ki > 10000 nM T64591 CW83DK 73213196 Ki = 501.19 nM T64591 CU3D9N 73388373 EC50 = 25118.86 nM T64591 C2E7QW 75201901 Ki = 7900 nM T64591 C8IDL3 75306277 Ki = 630.96 nM T64591 CM91EX 75965533 IC50 = 7 nM T64591 C92CDV 76309734 Ki = 7.3 nM T64591 C4WIP7 76309735 Ki = 1.6 nM T64591 C9DKY0 76309736 Ki = 208 nM T64591 CIO15U 76309745 Ki = 3.9 nM T64591 C3ZVG7 76309746 Ki = 35.3 nM T64591 CKI4L6 76309747 Ki = 72.2 nM T64591 CB12WY 76313417 Ki = 142 nM T64591 CEWV87 76313418 Ki = 1.2 nM T64591 CXT0N2 76313431 Ki = 316.23 nM T64591 CK9U0D 76313435 Ki = 73.8 nM T64591 C9Q5IC 76313436 Ki = 58.5 nM T64591 CM2A8D 76313437 Ki = 92.6 nM T64591 C5CEP8 76313438 Ki = 16.5 nM T64591 CMF40L 76313439 Ki = 14.9 nM T64591 C4B5GL 76313440 Ki = 18 nM T64591 C7B3MD 76313441 Ki = 40.4 nM T64591 CT72QD 76316931 Ki = 1.6 nM T64591 C67ZDO 76316932 Ki = 1.1 nM T64591 CA6O0D 76316934 Ki = 157 nM T64591 CHT0V4 76316950 Ki = 3.5 nM T64591 C2XM9Q 76316951 Ki = 15.1 nM T64591 CF9ME2 76316952 Ki = 16.3 nM T64591 CKB7Q3 76316953 Ki = 94.9 nM T64591 CS2Z7V 76320660 Ki = 199 nM T64591 CO04KJ 76320661 Ki = 8.7 nM T64591 CCMW30 76320680 Ki = 40 nM T64591 C2URV9 76320681 Ki = 4.6 nM T64591 C2Z4UE 76320682 Ki = 2 nM T64591 CJNA64 76320683 Ki = 37.3 nM T64591 CH9CV7 76324305 Ki = 1.9 nM T64591 CRYG31 76324319 Ki = 2.8 nM T64591 C41IFW 76327858 Ki = 1.89 nM T64591 C2HCL6 76327886 Ki = 8.3 nM T64591 CJ9Q6C 76327887 Ki = 18.8 nM T64591 C6F4DH 76331534 Ki = 5 nM T64591 CVHU83 76331535 Ki = 1 nM T64591 COS3V5 76335132 Ki = 0.9 nM T64591 C15HWF 76335133 Ki = 6300 nM T64591 CUS45K 76335134 Ki = 1300 nM T64591 C62UCI 76335155 Ki = 59.4 nM T64591 C0XY6P 76663424 IC50 = 58000 nM T64591 CWFN43 76800974 IC50 = 35 nM T64591 C70ZVB 86221574 Ki > 10000 nM T64591 CJ4A6R 87125710 IC50 = 7300 nM T64591 CP9IK4 87125800 IC50 = 21 nM T64591 CY2C6L 87403414 IC50 = 480 nM T64591 C2BM9L 89768534 IC50 = 1600 nM T64591 CB4Y7R 89768546 IC50 = 1500 nM T64591 CWG9T3 89940021 IC50 = 950 nM T64591 CKI70A 89943585 Ki = 560 nM T64591 CE6R1X 89943698 Ki = 440 nM T64591 C3EKN1 89943828 Ki = 3 nM T64591 C8ASH6 89943878 Ki > 1000 nM T64591 CH21GZ 89943908 Ki = 3 nM T64591 C9MG8P 90022612 IC50 > 100000 nM T64591 C2HUL4 90659973 Ki > 100000 nM T64591 CKM05S 90664904 IC50 > 100000 nM T64591 CEMZ15 118464420 Ki > 10000 nM T64591 CV2L6O 118464425 Ki > 10000 nM T64591 CFNG86 118464427 Ki > 10000 nM T64591 CUOQ12 121320365 IC50 = 10400 nM T64591 C4A3VY 121320367 IC50 = 11 nM T64591 CL60XN 121320376 IC50 = 13000 nM T64591 CYN0Q7 121320378 IC50 = 11 nM T64591 CT91EQ 121320401 IC50 = 6 nM T64591 CQJ2H8 121320430 IC50 = 13 nM T64591 CHQU84 121320526 IC50 = 660 nM T64591 C1FPG7 121320536 IC50 = 9700 nM T64591 CYQ68E 121320543 IC50 = 17 nM T64591 C0S5AU 121327773 IC50 = 43 nM T64591 CM7JS3 121327774 IC50 = 15 nM T64591 C6WFA4 121327777 IC50 = 4 nM T64591 C7K8VS 121327805 IC50 = 11 nM T64591 C94WSM 121327812 IC50 = 7 nM T64591 C7ODW3 122195524 Ki > 900 nM T64591 CCK1L8 122553340 Ki = 52 nM T64591 CKDM68 123133764 EC50 > 25000 nM T64591 C4QM2E 124247485 Ki > 10000 nM T64591 C50GOC 130442480 Ki = 9100 nM T64591 CM04RF 130442572 Ki = 9300 nM T64591 CAVB41 132584404 Ki > 10000 nM T64591 CSV59E 134131673 IC50 = 4000 nM T64591 CHB9W4 134132108 IC50 = 22000 nM T64591 CL3IE5 134132150 IC50 = 5600 nM T64591 C9ARP8 134132529 IC50 = 1600 nM T64591 CI96JM 134132991 IC50 = 27000 nM T64591 CA4X5H 134133656 IC50 = 7 nM T64591 C6XCO7 134134094 IC50 = 690 nM T64591 CDSM51 134134865 IC50 = 320 nM T64591 CKB5T2 134136620 IC50 = 86000 nM T64591 C3GH1V 134136714 IC50 = 28000 nM T64591 C0JKY3 134138261 IC50 = 19000 nM T64591 C03MJH 134139949 IC50 = 87000 nM T64591 C1E2RC 134141899 IC50 = 50 nM T64591 CNK1L0 134142616 IC50 = 7 nM T64591 CXQ84A 134143789 IC50 = 12000 nM T64591 CS8D9B 134145411 IC50 = 9100 nM T64591 C7AU1K 134146761 IC50 = 4200 nM T64591 CBU81N 134149168 Ki > 10000 nM T64591 CD24RC 134150057 IC50 = 5 nM T64591 CH32TG 134153963 IC50 = 250 nM T64591 CXT4U8 134154132 IC50 = 230 nM T64591 CJ3HP6 134154444 IC50 = 11 nM T64591 CJZ1P5 134154585 IC50 > 97000 nM T64591 CA5O8R 134154723 IC50 = 35 nM T64591 CT8XH7 134155582 IC50 = 13 nM T64591 CFY28D 134155678 IC50 = 29000 nM T64591 CKB4X1 134157219 IC50 = 2200 nM T64591 CZ2MU7 134157292 IC50 = 8 nM T64591 CDP46I 134157329 IC50 = 19 nM T64591 CXK4Q1 134157457 IC50 = 41000 nM T64591 C1GY2T 135156251 EC50 > 10000 nM T64591 C6N8GM 135367405 Ki > 10000 nM T64591 C6LU0C 135367816 Ki = 303 nM T64591 CD2TH9 135367820 Ki = 703 nM T64591 C5AMD9 135367857 Ki = 420 nM T64591 C7PXV8 135399236 Ki = 46.77 nM T64591 C8WL0I 135449090 Ki = 1511 nM T64591 CJW1V9 135570464 Ki = 575.44 nM T64591 CJF0P1 135600051 IC50 = 24.6 nM T64591 CBKP12 135976297 Ki = 0.17 nM T64591 CSNG95 135976299 Ki = 279 nM T64591 C6A8WK 136002690 IC50 = 55.2 nM T64591 CUKO20 136020617 Ki > 10000 nM T64591 COF0U5 136020618 Ki > 10 nM T64591 CF89JI 136030596 Ki > 10000 nM T64591 CE8GB9 136030693 Ki > 10000 nM T64591 C65VFI 136030744 Ki > 10000 nM T64591 COIX80 136054961 Ki > 10000 nM T64591 CS0JL5 136118616 Ki = 5916 nM T64591 C8RH6M 136118617 Ki = 6178 nM T64591 C5UDW3 136118620 Ki = 656 nM T64591 C8I6UN 136118621 Ki = 1223 nM T64591 C0W1TM 136118658 Ki = 591 nM T64591 C40LYH 136118659 Ki = 2624 nM T64591 CAE39V 136188797 Ki > 10000 nM T64591 CLAP52 136259032 Ki > 10000 nM T64591 CX0LF6 137633214 IC50 > 10000 nM T64591 C93ZPK 137635141 IC50 = 440 nM T64591 CTU9Y7 137635902 IC50 = 150 nM T64591 C3UT9L 137643408 IC50 = 170 nM T64591 CVJ0Q7 137644763 IC50 = 39000 nM T64591 C9K7VP 137644928 IC50 = 120 nM T64591 CQ5H2Y 137645815 IC50 = 29 nM T64591 CV9T6B 137647317 IC50 = 25 nM T64591 C3Y2SW 137649484 IC50 = 150 nM T64591 C6RJ8V 137649905 IC50 = 23 nM T64591 CVON14 137654242 IC50 > 100000 nM T64591 CJC95L 137654434 IC50 > 10000 nM T64591 COVD20 137655697 IC50 = 9 nM T64591 C6CYW8 137657023 IC50 = 180 nM T64591 CS3K4D 137659736 IC50 = 190 nM T64591 CX39HQ 137659815 IC50 = 27 nM T64591 C4GOE0 137660090 IC50 = 6700 nM T64591 CP48RG 137660174 IC50 = 100 nM T64591 C0B6HQ 137660214 IC50 = 3.8 nM T64591 C3FZL5 141725921 IC50 = 710 nM T64591 C7KC3T 145963830 Ki = 860 nM T64591 CHDN35 145964150 Ki > 10000 nM T64591 C1KH2E 145964159 Ki = 240 nM T64591 C12OVL 145965034 Ki > 10000 nM T64591 C5W4LM 145965940 Ki = 1800 nM T64591 C81VUO 145967771 Ki > 10 nM T64591 CJS56K 145967795 Ki = 6700 nM T64591 C06AFP 145967982 IC50 = 9 nM T64591 CIN05D 145968525 IC50 = 1400 nM T64591 CQJ5O8 145971635 Ki > 10000 nM T64591 C79TNE 145972796 Ki = 3600 nM T64591 C6XIN0 145974114 Ki > 10000 nM T64591 CD8ZL6 145974750 Ki > 10 nM T64591 C6PH4F 145975226 Ki = 3100 nM T64591 C71CYU 145975946 Ki > 10000 nM T64591 C2TN8W 145976085 Ki = 150 nM T64591 C1G4TW 145976577 IC50 = 62 nM T64591 C6BFY7 145977338 Ki = 950 nM T64591 C0Y6QO 145977799 Ki = 77 nM T64591 C3BI1R 145978113 Ki = 6700 nM T64591 CMR64J 145978573 IC50 = 6 nM T64591 CQU8R0 145978665 Ki = 2800 nM T64591 C6AV9G 145978819 Ki > 10000 nM T64591 C86XQR 145988313 Ki > 10000 nM T64591 CSYV30 145991039 EC50 > 25000 nM T64591 CC2G1V 146025727 Ki = 7600 nM T64591 C6P3SR 153287553 Ki > 10000 nM T64591 CV9G7Z 153287572 Ki > 10000 nM T64591 CO85KL 153287574 Ki > 10000 nM T64591 CUSA24 155519891 Ki > 10000 nM T64591 CB79ZW 155536080 Ki > 10000 nM T64591 C3N9VU 10251906 Ki > 500 nM T64591 CB0LH8 11602721 IC50 = 25118.86 nM T64591 CTAK49 11660066 IC50 = 100000 nM T64591 CQ1LV7 135508617 Ki = 1000 nM T64591 CUZ1D8 44564663 IC50 = 50118.72 nM T64591 D00AVR 135476741 Ki = 3029 nM T64591 D00CRA 1574 Ki = 1200 nM T64591 D00OBS 44559159 Ki > 10000 nM T64591 D01FFX 24691160 Ki = 311 nM T64591 D01JXM 46222048 Ki > 1000 nM T64591 D02OYL 46831055 IC50 = 7900 nM T64591 D03HCT 25196629 IC50 = 2400 nM T64591 D03JPN 11173546 Ki = 150 nM T64591 D03TPY 9885123 Ki = 1.2 nM T64591 D04CUL 25196633 IC50 = 2000 nM T64591 D05YAR 2758 IC50 = 257039.58 nM T64591 D05ZUX 44207909 Ki >= 1000 nM T64591 D06EPZ 25196850 IC50 = 11600 nM T64591 D06QIQ 44592241 Ki = 404 nM T64591 D07ZZD 9794818 Ki = 13 nM T64591 D08BCF 5011 Ki = 3.7 nM T64591 D08JLW 119376 Ki > 10000 nM T64591 D08OFG 11177588 Ki > 10000 nM T64591 D08VGJ 9904281 Ki = 172 nM T64591 D09HJL 10331436 Ki > 10000 nM T64591 D0AJ3C 9819593 Ki = 5.012 nM T64591 D0B1KT 15953802 Ki = 100000000 nM T64591 D0C5RZ 5610 EC50 = 26000 nM T64591 D0C9TY 16727408 Ki = 2 nM T64591 D0CK9K 6918513 IC50 > 1000 nM T64591 D0F6CD 5202 EC50 = 141 nM T64591 D0FF6S 16038374 IC50 > 10000 nM T64591 D0G2BS 5013 Ki = 0.4571 nM T64591 D0G7QT 10131112 IC50 = 34 nM T64591 D0I4BZ 6604914 Ki = 0.182 nM T64591 D0K9NK 16066792 IC50 = 4800 nM T64591 D0L5MW 181743 Ki > 10000 nM T64591 D0P2HR 3510 Ki = 1.45 nM T64591 D0QM9Y 25196851 IC50 = 5700 nM T64591 D0S0XK 9863146 IC50 = 1.413 nM T64591 D0SA4A 1354 EC50 = 3800 nM T64591 D0T2RY 9948320 Ki >= 1000 nM T64591 D0V9CG 44422402 IC50 = 7500 nM T64591 D0W8EP 5191 Ki = 125.89 nM T64591 D0X3HB 25196630 IC50 = 1900 nM T64591 D0X5DC 6549 IC50 = 141253.75 nM T64591 D0X7HD 11184481 IC50 = 5 nM T64591 D0Y4WI 44422187 IC50 = 13600 nM T64591 D0Y9TL 13702393 Ki = 1051 nM T64591 D0Z4JL 25196743 IC50 = 3300 nM T50973 D0P1BE 24812126 IC50 = 4000 nM T50973 C34OEY 21356 IC50 = 6 nM T50973 C1S7MV 127868 IC50 = 900 nM T50973 C5OYF0 277922 IC50 = 340 nM T50973 CWMS43 805922 IC50 = 6309.57 nM T50973 CB6U7D 822958 IC50 = 1700 nM T50973 C4YS6W 2757392 IC50 = 79.43 nM T50973 CG25PE 2795549 IC50 = 16700 nM T50973 CI4W2F 2795575 IC50 = 990 nM T50973 CBL62V 3067254 IC50 = 3300 nM T50973 CIF61J 4396579 IC50 = 12.59 nM T50973 CFE0S2 5282337 IC50 = 37 nM T50973 C94OHV 9816607 IC50 = 20 nM T50973 C6OV7P 9859947 IC50 = 20 nM T50973 CF5K2A 9926280 IC50 = 200 nM T50973 C5TC4S 9949670 IC50 = 180 nM T50973 CIC2L0 12582972 IC50 = 38 nM T50973 C5ND4C 13337779 IC50 = 100 nM T50973 CJD2K1 13337784 IC50 = 3162.28 nM T50973 CFQ70N 16636975 IC50 = 5011.87 nM T50973 CBAR18 22411571 IC50 = 1300 nM T50973 CA4GV8 23445016 IC50 = 3.2 nM T50973 CDK09S 23445120 IC50 = 90 nM T50973 C3VX5A 24277353 IC50 = 12 nM T50973 CX2KA9 24812233 IC50 = 39000 nM T50973 CDC2H6 43163556 IC50 = 125.89 nM T50973 CQ98VG 44632789 IC50 = 6510 nM T50973 CQVL20 44632916 IC50 > 10000 nM T50973 C71ILX 44632919 IC50 = 0.5 nM T50973 C7FC5Q 44633034 IC50 = 0.6 nM T50973 CGW7M3 44633035 IC50 = 19 nM T50973 C82SUZ 44633152 IC50 = 32 nM T50973 C40CIT 44633259 IC50 = 22 nM T50973 CRMB86 44633501 IC50 = 76 nM T50973 C9GWV5 44633650 IC50 = 0.2 nM T50973 C9D2RK 44633929 IC50 = 17 nM T50973 C71PCD 50972207 IC50 = 1700 nM T50973 CPHR01 53328211 IC50 = 2 nM T50973 C8SPK7 53329674 IC50 = 2300 nM T50973 CVI5T8 53329675 IC50 > 10000 nM T50973 C6S7IH 53330015 IC50 = 5060 nM T50973 CUP4M7 53330366 IC50 > 10000 nM T50973 C8JB4H 53330367 IC50 > 10000 nM T50973 C3FU4W 53330702 IC50 > 10000 nM T50973 C81IAD 53330703 IC50 > 10000 nM T50973 CSZO84 57296890 IC50 > 10000 nM T50973 C65CUS 57569654 IC50 = 990 nM T50973 C6G1BR 58367510 IC50 = 6 nM T50973 CCD63A 66817090 IC50 = 2130 nM T50973 C47TLX 67218051 IC50 = 38 nM T50973 CS26LT 67218064 IC50 = 0.9 nM T50973 C31GNA 67218312 IC50 = 0.3 nM T50973 CXE98L 67218371 IC50 = 5 nM T50973 CV51IA 67218427 IC50 = 1.2 nM T50973 C9LQR2 67218711 IC50 = 270 nM T50973 CLX7G3 67218735 IC50 = 0.7 nM T50973 CAY4H9 67325961 IC50 = 4000 nM T50973 C7PR9B 71282544 IC50 = 60 nM T50973 C4EVF3 71282597 IC50 = 64 nM T50973 C1XPD8 71282611 IC50 = 6 nM T50973 CHT23B 71282615 IC50 = 2 nM T50973 CKEH61 71282620 IC50 = 2.1 nM T50973 CC9Z4O 71282637 IC50 = 1740 nM T50973 CFMN98 71282644 IC50 = 0.5 nM T50973 CTJG35 71282673 IC50 = 0.3 nM T50973 CV7Z9D 71282689 IC50 = 350 nM T50973 CI9D7E 71282707 IC50 = 49 nM T50973 CU3I8P 71282725 IC50 = 40 nM T50973 CR04LD 71282761 IC50 = 0.9 nM T50973 CC38UG 71282784 IC50 = 83 nM T50973 CP1LN0 71282789 IC50 = 11 nM T50973 CB85NC 71282795 IC50 = 33 nM T50973 CU5L0Z 71282803 IC50 = 2130 nM T50973 CW4P0M 71282805 IC50 = 25 nM T50973 CQ5S6M 71282822 IC50 = 260 nM T50973 C0E9KZ 71282844 IC50 = 12 nM T50973 CIXJ40 71292353 IC50 = 2050 nM T50973 CRH19K 71292530 IC50 > 10000 nM T50973 CL6U3P 71292547 IC50 = 270 nM T50973 C8AKS4 82018077 IC50 = 50.12 nM T50973 C1SN7Q 82388114 IC50 = 1.5 nM T50973 CI46SG 82661260 IC50 = 0.3 nM T50973 C7UNS0 82663512 IC50 = 19 nM T50973 C46LFP 83756696 IC50 = 630.96 nM T50973 C1JX5L 83758092 IC50 = 1000 nM T50973 CTZL06 83820048 IC50 = 340 nM T50973 CRV51S 84018322 IC50 > 6309.57 nM T50973 CHX41G 84672230 IC50 = 3162.28 nM T50973 C5GWA7 84689388 IC50 = 1000 nM T50973 CGS34E 84700879 IC50 = 1995.26 nM T50973 CYO86V 84712290 IC50 = 39.81 nM T50973 CE0SO2 84789826 IC50 > 10000 nM T50973 CR51GB 91810763 IC50 = 125.89 nM T50973 C4HZG2 91810764 IC50 = 3.981 nM T50973 CC5N0T 95486126 IC50 = 9500 nM T50973 C61ICW 105539874 IC50 = 6.31 nM T50973 CVD41N 116899728 IC50 = 1.2 nM T50973 CK37QI 116899750 IC50 = 76 nM T50973 CMO2D3 116899761 IC50 = 0.9 nM T50973 CO13LQ 116900901 IC50 = 4000 nM T50973 CLR9X1 117523700 IC50 = 0.2 nM T50973 CL17UV 117683501 IC50 > 10000 nM T50973 CZ9PD4 118174579 IC50 = 12.59 nM T50973 CWSY96 118174585 IC50 = 12.59 nM T50973 C3S8QK 118174598 IC50 = 25.12 nM T50973 C97DCM 118174599 IC50 < 794.33 nM T50973 CRN49G 118174612 Ki = 1 nM T50973 C7T1VE 118174613 IC50 = 10 nM T50973 CPY4E2 118174622 IC50 = 100 nM T50973 CE27ZT 118174645 IC50 = 5.012 nM T50973 CF5T1V 118174652 IC50 = 3.162 nM T50973 CFW23X 118174669 IC50 = 79.43 nM T50973 CP61WF 118174672 IC50 < 794.33 nM T50973 C7EZT6 118174704 IC50 = 12.59 nM T50973 CFAI95 118174706 IC50 = 3.162 nM T50973 C6L1GX 118174709 IC50 = 316.23 nM T50973 CR72KZ 118174712 IC50 = 5011.87 nM T50973 C83RUW 118174714 Ki = 0.1 nM T50973 CJD39W 118174719 IC50 = 31.62 nM T50973 C7L0HO 118174738 IC50 < 794.33 nM T50973 CQK57J 118174786 IC50 = 1584.89 nM T50973 CH2T9E 118730424 IC50 = 1300 nM T50973 CX7JI1 118730425 IC50 = 140 nM T50973 C3HW9B 118730426 IC50 = 1500 nM T50973 CA63XP 118730427 IC50 = 430 nM T50973 CHUD20 118730428 IC50 = 37 nM T50973 CY68QF 118753129 IC50 = 17000 nM T50973 CV6Y2W 121415041 IC50 = 3.162 nM T50973 CW4AZ2 121415048 IC50 = 1.995 nM T50973 CZA48U 121415134 Ki = 0.05 nM T50973 C59XOU 122651968 IC50 = 251.19 nM T50973 C6BL5N 122651971 IC50 = 2.512 nM T50973 CO48CJ 124093262 IC50 = 1.995 nM T50973 C4E9JT 130136116 IC50 = 11 nM T50973 C4DR5M 131479729 IC50 = 17 nM T50973 CWER47 134131828 IC50 = 57 nM T50973 CC5D7S 134132839 IC50 = 60 nM T50973 CGV73C 134135607 IC50 = 2050 nM T50973 CB5F2G 134136793 IC50 = 0.3 nM T50973 C1F3TU 134137744 IC50 = 49 nM T50973 C0JZ1F 134137782 IC50 = 0.9 nM T50973 C9W0PX 134138153 IC50 = 83 nM T50973 C2PFT6 134138586 IC50 = 0.2 nM T50973 C4GT3S 134141064 IC50 = 2 nM T50973 CDOU02 134142257 IC50 = 2.1 nM T50973 C96LOG 134143276 IC50 = 550 nM T50973 COIL67 134144301 IC50 = 12 nM T50973 C4ILM6 134146801 IC50 = 38 nM T50973 CU20IF 134146980 IC50 = 6510 nM T50973 CLXI98 134147961 IC50 = 0.7 nM T50973 CMV4C0 134148848 IC50 = 5 nM T50973 CU87QH 134149072 IC50 = 12 nM T50973 C01TNQ 134150872 IC50 = 6 nM T50973 CW67AF 134151332 IC50 = 22 nM T50973 CDP5W2 134152168 IC50 = 9500 nM T50973 C6ERT4 134152894 IC50 = 430 nM T50973 CDCA87 134154503 IC50 = 32 nM T50973 C2Y9XD 134155572 IC50 = 0.5 nM T50973 CG2S1X 136067672 IC50 = 12 nM T50973 CA3M0L 137631488 IC50 = 2511.89 nM T50973 C8I1CO 137634379 IC50 = 1.585 nM T50973 C1HC7K 137634912 IC50 = 12.59 nM T50973 CZJ26T 137636219 IC50 = 501.19 nM T50973 CLV5W3 137637022 IC50 = 100 nM T50973 C0XZY7 137637142 IC50 = 5.012 nM T50973 C4EF2K 137637394 IC50 = 63.1 nM T50973 C5JA0Z 137638082 IC50 = 3.981 nM T50973 CC61OY 137638415 IC50 = 5.012 nM T50973 CQ1EJ8 137639644 IC50 = 5.012 nM T50973 CUA68W 137640130 IC50 = 2511.89 nM T50973 C5WM2X 137640576 IC50 = 3.162 nM T50973 CYF4V5 137642680 IC50 = 3.162 nM T50973 CT4E6H 137645014 IC50 = 5.012 nM T50973 C8VZX9 137646455 IC50 = 794.33 nM T50973 CZ1U8X 137648834 IC50 = 25.12 nM T50973 CG7YJ6 137649322 IC50 = 2.512 nM T50973 C5RYS1 137649485 IC50 = 39.81 nM T50973 C72OGI 137649940 IC50 = 3.162 nM T50973 CMT58V 137650016 IC50 = 5011.87 nM T50973 CPKS12 137650689 IC50 = 630.96 nM T50973 CXF13T 137652279 IC50 = 3.981 nM T50973 C10FQI 137655344 IC50 = 3.162 nM T50973 COS58X 137658639 IC50 = 5.012 nM T50973 CG2F3P 137660909 IC50 = 3.162 nM T77613 D06BCB 443955 IC50 > 10000 nM T77613 D03GTM 118485599 IC50 = 1000 nM T77613 D0J1LK 118485649 IC50 = 53 nM T77613 D0WS3T 72706254 IC50 = 26 nM T77613 C1B6ZL 662965 IC50 > 50000 nM T77613 C8JLO0 2243267 IC50 = 460 nM T77613 CMK39Q 10553487 IC50 = 48 nM T77613 C1B4XD 11992634 IC50 > 2000 nM T77613 CPX16N 11993169 IC50 > 2000 nM T77613 CW96SI 23624262 IC50 > 1000 nM T77613 C9WGI4 24802717 IC50 > 5000 nM T77613 C6EQG2 24963293 IC50 > 2000 nM T77613 CICF39 42629702 IC50 > 10000 nM T77613 CM3X9S 42629827 IC50 > 1000 nM T77613 CQN26J 42629945 IC50 > 5000 nM T77613 C6O5FX 42630062 IC50 > 10000 nM T77613 C71ZNR 42630180 IC50 > 5000 nM T77613 C4RHY0 42630191 IC50 > 10000 nM T77613 CT6RS9 42630192 IC50 > 10000 nM T77613 CYZL43 42630317 IC50 > 10000 nM T77613 CH42OZ 42630318 IC50 > 10000 nM T77613 C7X5AH 42630437 IC50 > 10000 nM T77613 CQU19I 44180409 IC50 = 21 nM T77613 CZJN98 46180643 IC50 = 35 nM T77613 CHA5Z0 49821469 IC50 > 1000 nM T77613 C1AYP0 49821627 IC50 > 500 nM T77613 C85AXR 49821714 IC50 > 1000 nM T77613 C6R4YN 50993785 IC50 = 10000 nM T77613 C0M6XL 50993786 IC50 = 10000 nM T77613 CGF65A 54670110 IC50 > 30000 nM T77613 C90ZLC 54670399 IC50 = 503 nM T77613 C4TGL7 56648496 IC50 > 1000 nM T77613 CH6C3L 56648679 IC50 > 10000 nM T77613 CCY79V 56648680 IC50 > 10000 nM T77613 CNE96P 56648857 IC50 > 5000 nM T77613 CX86AQ 56648859 IC50 > 5000 nM T77613 C0YD3P 56928304 IC50 > 5000 nM T77613 C8RO6A 56929788 IC50 > 1000 nM T77613 CD52CA 57391118 IC50 > 2000 nM T77613 C4XMB6 58547809 IC50 > 30000 nM T77613 CEB3G9 58547814 IC50 = 3680 nM T77613 C08QVG 58547833 IC50 = 8040 nM T77613 CFVG67 58547863 IC50 = 7920 nM T77613 CYZA38 58548077 IC50 = 7610 nM T77613 CN57ZH 67426178 IC50 > 10000 nM T77613 CY8J3O 68181896 IC50 > 30000 nM T77613 CUGH78 68654838 IC50 = 2511.89 nM T77613 C9GR3L 71153436 IC50 = 4900 nM T77613 C4GNJ3 71598545 IC50 > 1000 nM T77613 C68SDB 71719394 IC50 = 3981.07 nM T77613 CZ0G2X 72165213 IC50 > 10000 nM T77613 CQ3GD7 72704434 IC50 = 0.058 nM T77613 CPIO30 72706193 IC50 = 41 nM T77613 C1CQG9 72706253 IC50 = 3 nM T77613 CF4W8Z 72706442 IC50 = 27 nM T77613 C9JE6M 75815419 IC50 = 9.1 nM T77613 C52BXE 86705377 IC50 = 190 nM T77613 CJ0ET7 90445922 IC50 = 4 nM T77613 C1JPD6 91844700 IC50 = 6600 nM T77613 CYQV05 92471958 IC50 = 300 nM T77613 CYQ74R 118479645 IC50 > 10000 nM T77613 C0KPH4 118485600 IC50 = 210 nM T77613 C43GZF 118485601 IC50 = 150 nM T77613 C8UT1Z 118485623 IC50 = 31 nM T77613 CC94IQ 118485651 IC50 = 11 nM T77613 CLN89E 122184999 IC50 = 230 nM T77613 CK0TQ8 122185000 IC50 = 83 nM T77613 C8ZLF7 122185001 IC50 = 22 nM T77613 CV65IM 122185002 IC50 = 8 nM T77613 C4FQX3 122185003 IC50 = 38 nM T77613 CEXL86 122185006 IC50 = 70 nM T77613 CRJE23 122185011 IC50 = 2.4 nM T77613 CZ2HE3 122185012 IC50 = 458 nM T77613 CL89YP 122220126 IC50 = 4.5 nM T77613 CVX7U9 127029185 IC50 = 2629 nM T77613 C4UR7D 127038167 IC50 > 1000 nM T77613 C4H2TJ 127038168 IC50 > 1000 nM T77613 CL9JT8 127038169 IC50 > 1000 nM T77613 CJPX60 127038509 IC50 > 1000 nM T77613 C26EAG 127038511 IC50 > 1000 nM T77613 CTM9E4 127038512 IC50 > 1000 nM T77613 C6AQ2U 127038513 IC50 > 1000 nM T77613 CV1FM0 127038868 IC50 > 1000 nM T77613 CADU23 127038869 IC50 > 1000 nM T77613 CACJ46 132489333 IC50 > 10000 nM T77613 CZ09EG 135418212 IC50 = 38 nM T77613 C7GC0D 135436665 IC50 > 10000 nM T77613 C3R8SE 135457869 IC50 = 4950 nM T77613 CWQG94 135484473 IC50 = 2650 nM T77613 C2E3GU 135541419 IC50 = 50 nM T77613 C9IJK1 135566935 IC50 = 473 nM T77613 CX7I5Z 135721222 IC50 = 2630 nM T77613 CTX54Z 135896326 IC50 = 9800 nM T77613 CH6QL0 136059722 IC50 = 7810 nM T77613 C2J7ZU 136059723 IC50 > 10000 nM T77613 CN06GO 136059724 IC50 > 10000 nM T77613 C8EA6G 136059725 IC50 > 10000 nM T77613 C31KAG 136059726 IC50 > 10000 nM T77613 C12UMG 136059728 IC50 > 10000 nM T77613 CRP24A 136087045 IC50 = 2300 nM T77613 C7SUX4 136087050 IC50 = 1900 nM T77613 C8UF7G 136087052 IC50 = 18000 nM T77613 C8TQ7A 136217455 IC50 = 18000 nM T77613 C0YMI5 137631826 IC50 = 150 nM T77613 C6KYD7 137700754 IC50 = 1300 nM T77613 CM3UF7 137700779 IC50 > 20000 nM T77613 CPTE92 138319693 IC50 > 32000 nM T77613 C4W2YJ 145961173 IC50 = 596 nM T77613 C81NCL 145962793 IC50 = 52 nM T77613 CA80PU 145962849 IC50 = 27 nM T77613 CHJ79V 145997874 IC50 > 10000 nM T77613 CADM48 155510637 IC50 = 1400 nM T77613 CT5EQ7 155511060 IC50 = 2400 nM T77613 CV0Y5H 155512206 IC50 = 2000 nM T77613 CHPM03 155517492 IC50 = 7800 nM T77613 CGLS24 155521088 IC50 = 1800 nM T77613 CYI51O 155523485 IC50 = 1400 nM T77613 C9CYA3 155525884 IC50 = 700 nM T77613 CQ7IJ0 155531325 IC50 = 2200 nM T77613 C07WDO 155532938 IC50 = 1200 nM T77613 C0M2UC 155539455 IC50 = 10000 nM T77613 C3KE9M 155548362 IC50 = 1700 nM T77613 CQ5P0M 155553114 IC50 > 10000 nM T77613 CX6F2U 155559756 IC50 = 1200 nM T56057 D00SUC 74766595 IC50 = 2300 nM T56057 D09NCT 53392492 IC50 = 3100 nM T56057 CWJ0U1 5312 IC50 = 16500 nM T56057 C06WZQ 222878 IC50 > 100000 nM T56057 COS62U 245007 IC50 > 100000 nM T56057 C0MHV8 252439 IC50 = 1100 nM T56057 C5K3ZJ 459531 IC50 = 63095.73 nM T56057 C2OS3W 2238068 IC50 > 100000 nM T56057 CEQ4V8 2723716 IC50 > 100000 nM T56057 CTC90M 6519698 IC50 = 794.33 nM T56057 CCYF63 9942424 IC50 = 10000 nM T56057 CF47JU 25138011 IC50 = 11200 nM T56057 CU8AX0 55281807 IC50 = 98000 nM T56057 C6QTC3 64393791 IC50 = 39810.72 nM T56057 CM9Y5X 64394359 IC50 > 100000 nM T56057 CELF46 64394751 IC50 = 1258.93 nM T56057 C8K7LG 64395323 IC50 = 3981.07 nM T56057 CL3HT1 71449736 IC50 = 41700 nM T56057 CJH86V 71451542 IC50 > 100000 nM T56057 CH38AO 71453382 IC50 > 100000 nM T56057 C2U4AQ 71458738 IC50 > 100000 nM T56057 C5XA3R 71733941 IC50 = 9500 nM T56057 C4PW1L 71734037 IC50 = 7300 nM T56057 C6GDP2 71765680 IC50 = 794.33 nM T56057 CN53LH 71765996 IC50 = 630.96 nM T56057 C2RT5O 71765999 IC50 > 100000 nM T56057 COCF38 71767872 IC50 = 2511.89 nM T56057 CYF8O7 71767874 IC50 = 6309.57 nM T56057 C68RKH 76310231 IC50 = 27000 nM T56057 CO1EN3 76317452 IC50 = 2700 nM T56057 CT5FZ8 76321184 IC50 = 18000 nM T56057 C6XRT0 76321186 IC50 = 76000 nM T56057 CKB5O9 76328366 IC50 = 16000 nM T56057 CUNK03 76335652 IC50 = 14000 nM T56057 CX23ZP 78426670 IC50 > 2500 nM T56057 CMR52S 78426698 IC50 = 14300 nM T56057 CKXW73 78427224 IC50 > 2500 nM T56057 C9IMX6 81750118 IC50 = 3981.07 nM T56057 C63ATV 81750201 IC50 = 12589.25 nM T56057 CHY73I 81750365 IC50 = 1995.26 nM T56057 C69YUM 81751142 IC50 = 2511.89 nM T56057 CIG3E9 83672127 IC50 > 100000 nM T56057 C17WNZ 83698744 IC50 > 100000 nM T56057 CRQ51Z 86346639 IC50 > 1000 nM T56057 C83TUW 89825693 IC50 = 5011.87 nM T56057 C2NA5I 91801131 IC50 > 100000 nM T56057 CP3DK0 96607511 IC50 = 1000 nM T56057 C10RDJ 101882871 IC50 > 100000 nM T56057 C86LNW 101882872 IC50 = 31622.78 nM T56057 C4FPD3 112726150 IC50 > 100000 nM T56057 C6YT2Q 118598059 IC50 > 4000 nM T56057 C8E2KI 122191450 IC50 = 39810.72 nM T56057 C75JVN 122191451 IC50 > 100000 nM T56057 C3YX7W 122191453 IC50 > 100000 nM T56057 C3IBR8 122191455 IC50 = 50118.72 nM T56057 C59KNQ 122191457 IC50 > 100000 nM T56057 CM5X8J 122191459 IC50 = 79432.82 nM T56057 C7ASR0 122191460 IC50 = 79432.82 nM T56057 CRI6J4 122191461 IC50 > 100000 nM T56057 CAS4H6 122191462 IC50 = 63095.73 nM T56057 C9J6LX 122191463 IC50 > 100000 nM T56057 C75NJO 122191464 IC50 = 39810.72 nM T56057 C50VYK 122191465 IC50 = 15848.93 nM T56057 CSKY20 122191466 IC50 > 100000 nM T56057 CS3L8H 122191467 IC50 > 100000 nM T56057 CZ2NV1 122191468 IC50 = 50118.72 nM T56057 CYTW93 122191469 IC50 = 63095.73 nM T56057 CZV45H 122191470 IC50 = 100000 nM T56057 CF6I2N 122191471 IC50 > 100000 nM T56057 CZU02B 122191472 IC50 > 100000 nM T56057 CE27AS 122191473 IC50 > 100000 nM T56057 CAJ28B 122191475 IC50 = 50118.72 nM T56057 C36PDK 122191476 IC50 = 79432.82 nM T56057 CQ04FW 122191477 IC50 = 100000 nM T56057 C12OHA 122191478 IC50 = 50118.72 nM T56057 CL2K0J 122191479 IC50 = 79432.82 nM T56057 CT6HG3 122191480 IC50 = 19952.62 nM T56057 CK7LD6 122191481 IC50 = 12589.25 nM T56057 CMJ72N 122191482 IC50 = 12589.25 nM T56057 C6H2YQ 122383780 IC50 = 106000 nM T56057 CT2UZ4 125377518 IC50 > 100000 nM T56057 CL9EY7 127025757 IC50 = 490 nM T56057 C2D9TW 127026045 IC50 > 20000 nM T56057 CDK5R4 127026046 IC50 = 270 nM T56057 CBA6Z7 127026047 IC50 = 1500 nM T56057 CC62IF 127026048 IC50 = 1300 nM T56057 C19AYI 127026049 IC50 = 1400 nM T56057 CPOS14 127026050 IC50 = 1200 nM T56057 CG9PV5 127027278 IC50 = 200 nM T56057 C56CWO 127027279 IC50 = 1200 nM T56057 C7TJA3 127028289 IC50 = 2600 nM T56057 CH4FB5 127028601 IC50 = 150 nM T56057 CUL8I7 127028602 IC50 = 750 nM T56057 C1NIW3 127028603 IC50 = 550 nM T56057 CUD41F 127028604 IC50 = 1000 nM T56057 CWBS06 127028605 IC50 = 740 nM T56057 CA59FE 127028621 IC50 > 20000 nM T56057 CL0G1Z 127028622 IC50 = 210 nM T56057 C3KS1F 127028624 IC50 = 2100 nM T56057 CGP90K 127028625 IC50 = 1400 nM T56057 C2ZPT4 127028626 IC50 = 10000 nM T56057 C8F7SL 127029208 IC50 = 2100 nM T56057 CKQ61A 127029209 IC50 = 600 nM T56057 C68BYS 127029210 IC50 = 900 nM T56057 CNB68L 127035152 IC50 = 940 nM T56057 C73QDL 127036632 IC50 = 6100 nM T56057 C8QF1P 127037026 IC50 = 2200 nM T56057 CPM4V3 127037028 IC50 = 5800 nM T56057 CVOB08 127037169 IC50 > 100000 nM T56057 CY94VI 127037632 IC50 = 990 nM T56057 CT4O5U 135567037 IC50 > 100000 nM T56057 CC4H1N 135567038 IC50 = 31000 nM T56057 CQBH95 135567040 IC50 > 100000 nM T56057 CP6IH9 135567041 IC50 = 27000 nM T56057 C8HMG2 135567042 IC50 = 16000 nM T56057 CL9ZD4 135567108 IC50 = 26300 nM T56057 C1VAI3 135567112 IC50 = 48500 nM T56057 CO1F4A 135567128 IC50 > 100000 nM T56057 CE1SW8 136053677 IC50 > 100000 nM T56057 CMW30T 136053680 IC50 > 100000 nM T56057 CNY5T7 136053684 IC50 > 100000 nM T56057 C2V6MX 136644692 IC50 > 100000 nM T56057 CYG29R 138393334 IC50 = 52410 nM T56057 CNG82D 138393336 IC50 = 90220 nM T56057 CALG25 142810739 IC50 = 1200 nM T56057 C4M1EO 155519111 IC50 > 100000 nM T56057 CP8K5E 155540290 IC50 = 23970 nM T56057 CIM7D4 155548682 IC50 > 50000 nM T56057 CFR06L 155551969 IC50 > 50000 nM T56057 C3SQ4A 155569285 IC50 = 32260 nM T56057 D07IOY 10365 IC50 = 31622.78 nM T56057 D08IZY 3080614 IC50 = 316.23 nM T56057 D0B2WZ 15331 IC50 > 100000 nM T56057 D0S3DD 56963315 IC50 = 16 nM T56057 D0X5US 459617 IC50 = 100 nM T52447 D0G7UX 5284373 Ki = 2.58 nM T52447 D0M2OY 53259809 Ki = 2900 nM T52447 CFN3W4 311007 Ki = 63000 nM T52447 C0ACT7 53261396 Ki = 4900 nM T52447 CBWK59 53321090 Ki = 12 nM T52447 CL68DM 67255983 Ki = 950 nM T52447 CDY9G3 81689780 Ki = 2600 nM T52447 CWT5K3 118943806 Ki = 1330 nM T52447 C6K7DX 121231453 Ki = 22000 nM T52447 CNT97E 121231455 Ki = 9100 nM T52447 C0JMA9 127046107 Ki = 99 nM T52447 CEJ50V 130476037 IC50 = 1500 nM T52447 CC93VW 130476052 IC50 = 44000 nM T52447 C3XK5M 130476228 IC50 = 54000 nM T52447 C4MKS5 130476248 IC50 = 10000 nM T52447 C43HFX 130476250 IC50 = 190 nM T52447 CJN5Y0 130476253 IC50 = 3600 nM T52447 CKO3R5 130476256 IC50 = 4 nM T52447 CI1U7H 130476269 IC50 = 4100 nM T52447 CDK68A 130476279 IC50 = 1700 nM T52447 CI0SD8 130476467 IC50 = 600 nM T52447 CT7RY9 130476468 IC50 = 2800 nM T52447 CO9NT0 130476469 IC50 = 490000 nM T52447 CDPO73 131971481 IC50 = 80000 nM T52447 CL6WM2 140430653 IC50 = 735 nM T52447 CGK8Q7 155512090 IC50 = 870000 nM T52447 CS0E5L 155521155 IC50 > 100000 nM T52447 CG7QZ0 155541962 IC50 = 1700 nM T52447 CJE72T 155544108 IC50 > 100000 nM T52447 CK3YR4 155545905 IC50 > 100000 nM T52447 C2I9SQ 155549580 IC50 = 3500 nM T52447 CH52ZB 155557873 IC50 > 30000 nM T52447 CWI30L 155569565 IC50 > 100000 nM T27812 D00TLN 2913 Ki = 4100 nM T27812 D01AXB 60835 Ki = 0.24 nM T27812 D01AZG 5073 Ki = 1400 nM T27812 D01JMC 11658860 Ki = 2606 nM T27812 D01UTL 2995 Ki = 20 nM T27812 D01ZII 2726 Ki = 63.1 nM T27812 D02PPN 4158 IC50 = 5100 nM T27812 D02XOK 6917779 IC50 = 320 nM T27812 D03WEX 9966051 Ki = 1.6 nM T27812 D04CRN 54841 IC50 = 48 nM T27812 D04XPW 446220 Ki = 45 nM T27812 D05GKD 33741 IC50 = 1900 nM T27812 D06GDY 43815 Ki = 0.04 nM T27812 D06ZUK 3696 Ki = 0.52 nM T27812 D07HQC 4236 Ki = 570000 nM T27812 D08RBC 146570 Ki = 1 nM T27812 D08VRO 3822 Ki > 10000 nM T27812 D09VGC 65833 Ki = 22 nM T27812 D0CQ0Z 33630 Ki = 1000 nM T27812 D0D1AL 3559 Ki = 1800 nM T27812 D0H3HM 60795 Ki = 31.62 nM T27812 D0H7KF 5002 Ki > 18000 nM T27812 D0H8QL 4020 Ki = 45 nM T27812 D0HQ6N 1201549 IC50 = 24100 nM T27812 D0J5RN 9690109 IC50 = 232000 nM T27812 D0K0TC 68617 IC50 = 3 nM T27812 D0O3FG 125017 Ki = 15 nM T27812 D0P1UX 5656 Ki = 11 nM T27812 D0R1JV 60854 Ki = 53 nM T27812 D0T2XU 4927 IC50 = 7590 nM T27812 D0T3LF 5826 EC50 = 1770 nM T27812 D0T7OW 681 IC50 > 30000 nM T27812 D0TR5X 3386 Ki = 0.72 nM T27812 D0V4QS 135398745 Ki > 15000 nM T27812 D0WY5Q 77991 IC50 > 1000 nM T27812 D0X4ZR 444 IC50 > 100 nM T27812 D0X6BV 6918314 IC50 = 0.4 nM T27812 D0X7DE 4449 Ki = 290 nM T27812 D0Y5DO 2771 Ki = 1.6 nM T27812 D0Y5UG 2160 Ki = 4.3 nM T27812 D0Z1RV 135398737 Ki = 3900 nM T27812 D0ZS8P 2801 Ki = 0.28 nM T27812 D00WLO 3455 IC50 = 73 nM T27812 D03QIE 47953 IC50 = 117 nM T27812 D04PXS 11658655 IC50 = 12.3 nM T27812 D07AHC 65650 IC50 = 5.9 nM T27812 D0DH5X 44472635 IC50 > 10000 nM T27812 D0F5NJ 1615 Ki = 0.73 nM T27812 D0I2XM 3038500 IC50 = 5000 nM T27812 D0J9PT 58212050 IC50 = 1.1 nM T27812 D0L9QM 59568713 IC50 = 120 nM T27812 D0LI1C 44469321 IC50 > 10000 nM T27812 D0WL3H 15983287 IC50 = 723 nM T27812 D0Y2GJ 44182694 Ki = 1.02 nM T27812 D00OWF 5280953 Ki > 10000 nM T27812 D01ESB 157918 Ki = 21 nM T27812 D01NJT 65856 Ki = 661 nM T27812 D02JMI 9888211 Ki = 0.7943 nM T27812 D06BPG 4528 Ki = 874 nM T27812 D06DZI 107780 IC50 = 1000 nM T27812 D07BCO 5684 IC50 > 4500 nM T27812 D0A5RD 9795056 IC50 = 387 nM T27812 D0G1RH 6918446 IC50 = 0.002 nM T27812 D0H9GQ 9795276 IC50 = 12 nM T27812 D0K9JP 9928332 Ki = 3.77 nM T27812 D0S6PJ 5012 Ki = 0.17 nM T27812 CLJ8R2 1576 EC50 = 3860 nM T27812 CAG0J1 5523 IC50 = 1493 nM T27812 C6YZ2N 8554 IC50 > 100000 nM T27812 CK9A6Z 9280 IC50 > 10000 nM T27812 C5H9CN 9287 Ki = 812 nM T27812 CRU9X7 16458 Ki > 10000 nM T27812 C32HPI 19026 IC50 = 550 nM T27812 C1VSC0 19027 IC50 > 1000 nM T27812 C3VL1J 27694 Ki = 46700 nM T27812 CGU3Z5 42145 Ki = 27000 nM T27812 CQR7U2 44024 Ki = 57 nM T27812 CD9E4R 44668 IC50 = 30 nM T27812 CVL6S2 44831 IC50 = 400 nM T27812 C6WDL7 49756 Ki > 10000 nM T27812 C0OST7 55993 Ki = 935 nM T27812 C6KXM1 62857 Ki = 1.1 nM T27812 C9E6LD 62923 IC50 = 200 nM T27812 CL5WD4 67786 Ki > 10000 nM T27812 CI6QK3 77250 Ki = 35000 nM T27812 C8X5YU 77251 Ki = 12600 nM T27812 C0O3IG 77252 Ki = 1160 nM T27812 C92HJY 77995 Ki = 0.78 nM T27812 CYKE31 104920 IC50 = 3840 nM T27812 CF65AM 107934 EC50 = 3162.28 nM T27812 C5Q1OD 108220 Ki = 29.17 nM T27812 C3ZFS8 122252 Ki = 1.4 nM T27812 C7B9PA 122501 Ki > 10000 nM T27812 C3FW1L 132499 IC50 = 177 nM T27812 CAR7Y4 146571 Ki = 1 nM T27812 CXUG79 148883 IC50 > 10000 nM T27812 C0ALO6 152215 IC50 = 690 nM T27812 C56XJT 157919 Ki = 21 nM T27812 CGT8R0 160510 Ki > 10000 nM T27812 CD1H4C 204666 Ki = 1760 nM T27812 CAW9K8 211262 Ki > 10000 nM T27812 CQ97NL 242919 Ki = 910 nM T27812 C1KUD9 264388 Ki > 10000 nM T27812 CR7MP9 264389 Ki > 10000 nM T27812 CQK09D 279413 Ki = 630 nM T27812 C2V5FA 398712 Ki = 200 nM T27812 CDR63W 403508 Ki = 11 nM T27812 CE3N8G 411735 Ki > 10000 nM T27812 CYV1R3 417052 Ki > 10000 nM T27812 C31JMB 449842 Ki = 1.82 nM T27812 CZ53QF 656832 Ki = 95 nM T27812 CXQ6U0 735755 IC50 > 10000 nM T27812 CZN6S9 743974 IC50 > 100000 nM T27812 C2CT0Y 818024 Ki = 0.27 nM T27812 CK65MQ 826771 IC50 = 40 nM T27812 CQ0DV9 1393540 IC50 = 33000 nM T27812 C47BIF 1394484 IC50 = 46000 nM T27812 C1YED3 2199935 Ki = 75 nM T27812 C9CH5B 2769362 Ki = 29 nM T27812 CH24PD 2801930 Ki = 83.43 nM T27812 CA3S7R 3022645 Ki = 9 nM T27812 CZ9SV5 3025846 Ki = 68 nM T27812 CUE91A 3055249 IC50 = 730 nM T27812 C9EF2P 3058416 IC50 = 1000 nM T27812 C58WXN 3061874 IC50 = 240 nM T27812 CK8F0T 3080846 IC50 = 7540 nM T27812 C9HJ3S 3302814 Ki = 0.33 nM T27812 C0YXV3 3676358 Ki > 10000 nM T27812 C56JID 3763575 Ki = 30.4 nM T27812 CYH1O6 3992724 Ki = 24 nM T27812 CF12IO 4141883 Ki = 1510 nM T27812 CB0G8U 4605800 Ki = 2.3 nM T27812 COC2V5 4913097 IC50 = 570 nM T27812 CI56AJ 5141361 Ki = 0.36 nM T27812 C3KY9U 6101829 EC50 = 25000 nM T27812 C5FUA2 6328322 Ki = 46700 nM T27812 C8ZK1O 6328354 Ki = 57 nM T27812 C0IHP9 6336338 Ki = 0.009 nM T27812 CY4GC1 6918635 IC50 = 42 nM T27812 CY70ST 9794826 IC50 > 10000 nM T27812 C2ICW4 9794964 Ki = 822 nM T27812 CDEL49 9795462 Ki = 116 nM T27812 C6XYV0 9795623 IC50 = 30 nM T27812 CR2JV1 9795977 Ki = 530 nM T27812 C5FJ4K 9798438 IC50 = 2 nM T27812 CPG3J9 9798864 IC50 = 254 nM T27812 C68UYJ 9801487 Ki = 31.62 nM T27812 CX7I8J 9802187 Ki = 0.1 nM T27812 C5Z2KM 9805944 Ki = 6.2 nM T27812 C1W2VB 9814248 IC50 = 34.8 nM T27812 CAD92E 9815159 IC50 = 3.27 nM T27812 CS7V4Z 9816172 IC50 = 1.1 nM T27812 C7PUZ1 9816962 Ki = 2149 nM T27812 CT7OD0 9817610 Ki > 100 nM T27812 CB8N5S 9817852 IC50 = 2830 nM T27812 CI4KO5 9819496 Ki = 55 nM T27812 C45QPU 9820163 Ki = 1.5 nM T27812 CS6KM1 9820536 IC50 = 305 nM T27812 CEPW14 9834659 IC50 = 71 nM T27812 C8AHK9 9834987 IC50 = 56.8 nM T27812 C0I4OX 9835259 IC50 = 2 nM T27812 C1FQ5A 9835490 IC50 = 37.5 nM T27812 CQPO85 9835750 Ki = 4.8 nM T27812 C56BKA 9836263 IC50 = 5 nM T27812 C3W2ZV 9836377 IC50 = 3.77 nM T27812 CM85OH 9836429 IC50 = 650 nM T27812 C3DN1P 9836520 IC50 = 4.7 nM T27812 CX8P7C 9837869 Ki = 767 nM T27812 CY7K5Z 9838051 Ki = 266 nM T27812 C1YLP0 9838350 Ki = 338 nM T27812 C0YI3N 9839972 IC50 = 15 nM T27812 C36NME 9842337 Ki = 387 nM T27812 C1LOQ2 9842682 Ki = 276 nM T27812 CS1ID2 9846928 IC50 = 407 nM T27812 CM13ZV 9856041 Ki > 10000 nM T27812 CS14HB 9859833 IC50 = 0.48 nM T27812 CRBW42 9861124 IC50 = 3.28 nM T27812 CC0SQ3 9862968 IC50 = 2170 nM T27812 CIXO17 9863396 IC50 = 444 nM T27812 C0IR5C 9864943 Ki = 4.1 nM T27812 C1ZB4W 9865652 Ki = 0.09 nM T27812 CHM4D6 9866320 IC50 = 145 nM T27812 C3KGX7 9867350 Ki = 1.4 nM T27812 CN9YD5 9868131 IC50 = 2 nM T27812 C2WB5T 9868306 Ki = 0.54 nM T27812 CQ4LC2 9872676 Ki = 1430 nM T27812 CEJP40 9878793 IC50 = 904 nM T27812 CKC50T 9878987 IC50 = 3 nM T27812 CR0EG2 9879772 IC50 = 8.72 nM T27812 CQJ5X2 9879974 IC50 = 6.22 nM T27812 C93WSM 9880323 IC50 = 99000 nM T27812 C01ABG 9881528 Ki = 118 nM T27812 CLSP49 9881709 IC50 = 10000 nM T27812 CCZ84V 9881969 Ki = 594 nM T27812 CHNC28 9882029 Ki = 287 nM T27812 CY6QX4 9882047 Ki = 81.7 nM T27812 C7KP4G 9882069 Ki = 52647 nM T27812 C8Q4OZ 9884474 Ki = 0.06 nM T27812 C9AZ6P 9884876 IC50 = 4 nM T27812 CW76OG 9885700 IC50 = 6.3 nM T27812 CBQ7Y3 9886288 Ki = 0.12 nM T27812 CN52BU 9887951 IC50 = 70 nM T27812 CE28TW 9900179 IC50 = 1 nM T27812 CM3L0I 9900725 IC50 = 1063 nM T27812 CZUM05 9900755 IC50 = 60 nM T27812 CCFR97 9903806 Ki = 2.8 nM T27812 CPH07N 9903956 Ki = 111 nM T27812 CYWQ50 9906447 Ki > 10000 nM T27812 CUEZ75 9908121 Ki = 5.9 nM T27812 CCM2Z0 9908126 IC50 = 1 nM T27812 CYZ5N4 9909089 Ki = 1.259 nM T27812 C1CSK2 9910220 IC50 = 991 nM T27812 CSKJ62 9910492 IC50 = 5 nM T27812 CL5W7J 9920766 IC50 > 70000 nM T27812 C5T7UK 9921294 IC50 = 44000 nM T27812 C9MDU2 9921865 IC50 = 2600 nM T27812 CQX6R9 9924713 IC50 = 3 nM T27812 CQF2X8 9925089 IC50 = 5.1 nM T27812 C5Y8PI 9925806 IC50 = 0.16 nM T27812 CID4Y2 9928432 IC50 = 28.1 nM T27812 C3RVK7 9928961 IC50 = 3 nM T27812 CQX4W1 9929572 Ki = 45 nM T27812 C10VOI 9930235 IC50 = 34 nM T27812 CGD46V 9930573 Ki = 0.097 nM T27812 CPYN79 9930791 IC50 = 5 nM T27812 C6AZ3X 9943908 IC50 > 100 nM T27812 CS58EO 9944019 IC50 = 23 nM T27812 CX3ZK9 9946374 IC50 = 29.6 nM T27812 CV1T2W 9947009 IC50 = 4.8 nM T27812 CH6IJ8 9947172 IC50 = 17.1 nM T27812 C7QFK2 9947230 IC50 = 2 nM T27812 C9U2AT 9947569 IC50 = 9 nM T27812 CPBQ94 9948049 IC50 = 3168 nM T27812 CM7J6H 9948700 IC50 = 1960 nM T27812 CAP9K6 9949231 IC50 = 867 nM T27812 C76NBU 9950374 Ki = 0.52 nM T27812 CXUC75 9950482 IC50 = 9.7 nM T27812 C5JI4O 9951619 IC50 = 9 nM T27812 C79VHZ 9952054 IC50 = 2.53 nM T27812 CMI58L 9956563 IC50 = 0.078 nM T27812 CL56QZ 9957437 Ki = 8.3 nM T27812 C1NPJ7 9965169 IC50 = 9.47 nM T27812 C3KTF6 9965610 IC50 = 19.3 nM T27812 C6K7YM 9965748 IC50 = 8 nM T27812 CY9Q2M 9966187 IC50 = 6700 nM T27812 C6CXJ3 9966330 IC50 = 2.5 nM T27812 C49MPX 9966437 IC50 = 2.36 nM T27812 CJ2DK6 9966438 IC50 = 8.9 nM T27812 C7ZK5J 9966516 IC50 = 70000 nM T27812 CC35UV 9966603 IC50 = 8.09 nM T27812 CX85DP 9969177 IC50 = 5 nM T27812 C6YD3U 9970217 IC50 = 170 nM T27812 CXQT95 9972472 IC50 = 4.3 nM T27812 CFZ9D7 9972515 IC50 = 1 nM T27812 COP08X 9972881 IC50 = 2010 nM T27812 CAPD80 9973018 IC50 = 15 nM T27812 CR5XJ2 9975609 Ki = 41.2 nM T27812 C2XG1I 9977716 Ki = 6.31 nM T27812 CPX92V 9979309 Ki = 19.95 nM T27812 CXCP15 9980795 Ki = 351 nM T27812 CIT79L 9992137 IC50 = 31 nM T27812 CQG25B 9993136 IC50 = 3.8 nM T27812 CS98RN 9994556 IC50 = 300 nM T27812 C2AW8E 9996581 IC50 = 2.5 nM T27812 C2PT6Y 9996683 IC50 = 10 nM T27812 C8A6EZ 10001971 Ki = 15.85 nM T27812 CJ95XF 10003490 Ki = 1400 nM T27812 CQL12P 10004545 Ki > 2000 nM T27812 CD9JO4 10015148 IC50 = 64 nM T27812 CWDU13 10015606 IC50 = 1.4 nM T27812 CJQ2H6 10015826 IC50 = 58 nM T27812 CHG91I 10017115 Ki = 1.04 nM T27812 CQHW51 10023176 Ki = 0.7943 nM T27812 CH6OC0 10024324 Ki = 16.75 nM T27812 CL06BD 10027543 Ki = 135 nM T27812 C52JBP 10028898 Ki = 5.4 nM T27812 CPG46C 10039026 IC50 = 7.3 nM T27812 CU9I4O 10040854 IC50 = 5.3 nM T27812 C2C1XS 10042602 IC50 = 260 nM T27812 C25WVJ 10047566 IC50 = 1 nM T27812 CF84QJ 10048342 Ki = 79.43 nM T27812 C5MQ9L 10060174 IC50 = 33 nM T27812 CR79GU 10061525 IC50 = 1.6 nM T27812 COZ94V 10062443 Ki = 1.12 nM T27812 C79GJK 10062560 Ki = 0.49 nM T27812 C1NOQ0 10066050 IC50 = 6.2 nM T27812 CIC0W2 10068815 Ki = 10 nM T27812 C9KWT3 10071738 Ki = 0.7943 nM T27812 C1J4YU 10072978 Ki = 530 nM T27812 CV6R2F 10073139 Ki = 0.1585 nM T27812 C1LN4V 10084648 Ki = 0.25 nM T27812 CO50KM 10085525 Ki = 1.89 nM T27812 C6L5KD 10086762 IC50 = 5160 nM T27812 CW7K1U 10086952 Ki = 1060 nM T27812 C5H3MJ 10090352 IC50 = 15 nM T27812 C6KY5X 10090661 Ki = 5 nM T27812 CPQD23 10096087 Ki = 85 nM T27812 COMZ02 10107774 IC50 = 570 nM T27812 CO1R2Q 10110820 IC50 = 5 nM T27812 CC15UG 10111229 Ki = 46.9 nM T27812 CINW17 10130931 Ki = 1220 nM T27812 C6N2TK 10131545 IC50 = 4.51 nM T27812 C80GWE 10132137 IC50 = 5370 nM T27812 CVZ3S9 10132138 IC50 = 14.1 nM T27812 C26HWK 10132572 IC50 = 21.8 nM T27812 CL50NI 10150457 IC50 = 120000 nM T27812 C13VPI 10198613 Ki = 1430 nM T27812 CM9CT0 10198980 Ki = 230 nM T27812 C4J6DM 10199240 Ki = 479 nM T27812 CMKB87 10200680 IC50 = 15 nM T27812 C46ECI 10216348 Ki = 101 nM T27812 CF9B2N 10220613 Ki = 121 nM T27812 CG32IU 10220615 Ki = 1750 nM T27812 CI8NQ2 10220697 Ki = 102 nM T27812 C8C6IY 10221010 IC50 = 0.32 nM T27812 CYAV42 10236153 Ki = 3900 nM T27812 C6HUY5 10238982 Ki = 198 nM T27812 C0NLA3 10243659 IC50 = 1.7 nM T27812 C2D4YM 10244152 Ki = 0.53 nM T27812 CMSE68 10245407 IC50 = 7.9 nM T27812 CG2B7I 10247701 IC50 = 1760 nM T27812 CI2BC9 10263646 IC50 = 8.5 nM T27812 C5P0UZ 10263960 IC50 = 5.1 nM T27812 CQ4M3F 10265481 Ki = 1.46 nM T27812 CRXC41 10265748 IC50 = 6.2 nM T27812 CNW1L9 10265758 IC50 = 292 nM T27812 CF2M9O 10268223 IC50 = 3.61 nM T27812 CR2J1V 10271949 Ki = 19.8 nM T27812 C5AX7N 10291757 Ki = 4.51 nM T27812 C5HI6T 10293752 IC50 = 9 nM T27812 CB4C9E 10313840 Ki = 3.58 nM T27812 CMI2Y9 10314525 IC50 = 5.3 nM T27812 C1Z8AO 10314993 IC50 > 2000 nM T27812 CA3E4W 10316297 IC50 > 10000 nM T27812 C0OJ2C 10319235 Ki = 2.512 nM T27812 C8TBD5 10319565 Ki = 1.4 nM T27812 CPH30X 10319737 Ki = 10 nM T27812 CKE53N 10320283 IC50 > 10000 nM T27812 CISG65 10323598 IC50 > 1000 nM T27812 C18HWI 10332943 IC50 = 3 nM T27812 C9A0UX 10333208 IC50 = 30 nM T27812 C1ML2Q 10333844 IC50 = 3 nM T27812 C58YJO 10334599 IC50 = 65 nM T27812 C7AY2L 10337564 IC50 = 2000 nM T27812 CXG6B1 10341129 Ki = 1.995 nM T27812 CTS16A 10354918 IC50 = 7 nM T27812 CUF4G8 10355130 Ki = 25 nM T27812 CO8YX5 10355636 IC50 = 260 nM T27812 CK1X4I 10356972 IC50 = 14 nM T27812 C1A0VI 10359867 Ki = 85 nM T27812 C92IVO 10360093 IC50 = 140 nM T27812 CA4R1B 10362715 Ki = 0.47 nM T27812 CRZ15J 10363398 Ki = 0.04 nM T27812 CSWC08 10364638 IC50 = 25 nM T27812 C3R7VI 10367506 Ki = 229 nM T27812 CG73OS 10369316 IC50 > 1000 nM T27812 CN1L4S 10377587 IC50 = 4.3 nM T27812 C2W5VG 10377918 IC50 = 3.7 nM T27812 CG7ZD8 10379775 IC50 = 110 nM T27812 C3V2KB 10379785 IC50 = 710 nM T27812 CX13CN 10381502 IC50 = 4962 nM T27812 C0XG9M 10387420 Ki = 0.7943 nM T27812 CWZ0P2 10400022 IC50 = 6.6 nM T27812 CN2O8Q 10400315 Ki = 1.59 nM T27812 CY43ZX 10401043 IC50 = 2.9 nM T27812 CEAN45 10402966 IC50 = 109 nM T27812 C02ZET 10403162 Ki = 650 nM T27812 CUGW61 10403428 IC50 = 534 nM T27812 CSN67Q 10404183 IC50 = 6.8 nM T27812 C7H5TA 10405063 IC50 = 6.5 nM T27812 C23LGF 10411109 Ki = 210 nM T27812 CI9ZQ8 10428183 IC50 = 13 nM T27812 CR8J7I 10432519 Ki = 500 nM T27812 CJH4C9 10437435 IC50 = 48 nM T27812 CRKC54 10439429 Ki = 7.9 nM T27812 CRDP26 10446476 IC50 = 10 nM T27812 C98SIQ 10446567 Ki = 1.1 nM T27812 CJE4W0 10447238 IC50 = 240 nM T27812 CE5K4I 10447533 Ki = 5.6 nM T27812 C7X4BM 10447912 IC50 = 1.6 nM T27812 CL65VJ 10450883 Ki = 390 nM T27812 C9WA5Q 10452875 Ki = 10 nM T27812 CFK16Y 10454806 Ki = 5.012 nM T27812 CYMS64 10454807 Ki = 1.259 nM T27812 C38VGA 10457264 IC50 = 10000 nM T27812 C6ACL8 10467104 IC50 = 3.3 nM T27812 CE9ML0 10467904 IC50 = 6.5 nM T27812 C0Z9QA 10469659 IC50 = 22 nM T27812 C5Q2IO 10472386 Ki = 64 nM T27812 C7KU1T 10472626 IC50 = 85 nM T27812 CSZ56B 10472714 Ki = 25.6 nM T27812 C5HDQ3 10476240 IC50 = 5848 nM T27812 CL63TF 10477223 Ki = 0.7943 nM T27812 C86GXB 10477812 Ki = 2200 nM T27812 CWY2J3 10478217 Ki = 1.585 nM T27812 CRZ59G 10479666 Ki = 230 nM T27812 CW81LP 10480357 Ki = 1.3 nM T27812 CXKM90 10502796 IC50 = 14 nM T27812 CF7B1H 10520686 Ki = 740 nM T27812 CX69HP 10525046 IC50 = 1860 nM T27812 CYP31J 10530932 IC50 = 3800 nM T27812 C7TX6Q 10543664 Ki = 13 nM T27812 CJ6P1Z 10544672 Ki = 91 nM T27812 C3DR1F 10551367 Ki = 890 nM T27812 C0US7T 10568696 Ki = 73 nM T27812 COA6T3 10570967 IC50 > 10 nM T27812 C4U6NW 10575012 Ki = 1150 nM T27812 C3CYF7 10575547 Ki = 114 nM T27812 CG85VM 10578117 IC50 = 900 nM T27812 CC12NB 10591764 Ki = 93 nM T27812 C5G1OF 10594234 IC50 = 21 nM T27812 CAGB14 10598649 Ki = 55 nM T27812 C5X7BD 10600871 IC50 > 1000 nM T27812 C6K7IB 10624680 IC50 = 4700 nM T27812 CQW4H8 10627068 IC50 > 10 nM T27812 C5R0MA 10627612 IC50 > 1000 nM T27812 C8L4AG 10640435 Ki = 44 nM T27812 C69FME 10640436 Ki = 200 nM T27812 C71KTR 10645578 IC50 = 49179 nM T27812 CCZU47 10663468 Ki = 16 nM T27812 C2P5WV 10666153 Ki = 287 nM T27812 CQ7V9F 10670209 IC50 > 10 nM T27812 CX12VM 10670307 Ki = 438 nM T27812 C0VWZ3 10672803 IC50 = 10657 nM T27812 C75AQY 10673854 IC50 > 1000 nM T27812 C5FY3Q 10688125 Ki = 1700 nM T27812 CU58VP 10691286 Ki = 180 nM T27812 CG0V7W 10693838 Ki = 1300 nM T27812 CRLX06 10697639 Ki = 1.5 nM T27812 C26VWI 10712698 Ki = 4700 nM T27812 C5G9PK 10718709 IC50 > 1000 nM T27812 CPO3J8 10734429 Ki = 130 nM T27812 C3I7ZE 10740824 Ki = 550 nM T27812 CDZT46 10741033 Ki = 500 nM T27812 CRP3D6 10765459 Ki = 523 nM T27812 CP1N4Y 10788455 Ki = 556 nM T27812 CGM3Q2 10788465 Ki = 125 nM T27812 C2Q4BI 10813108 Ki = 320 nM T27812 CNB26G 10813109 Ki = 87 nM T27812 C9M7UN 10835740 Ki = 1530 nM T27812 C0GX8V 10836499 Ki = 220 nM T27812 C1GAE4 10837110 Ki = 350 nM T27812 CAM8P0 10852732 Ki = 25 nM T27812 C5JU4D 10860718 Ki = 600 nM T27812 CDF36V 10890308 EC50 = 2137962.09 nM T27812 CMS0Z2 10893018 Ki = 224 nM T27812 C58SAQ 10904197 Ki = 5.5 nM T27812 CE9JL7 10934835 IC50 = 60 nM T27812 C9VH4C 10946580 Ki = 1.94 nM T27812 CUG82R 10993971 Ki = 164 nM T27812 C15TXK 10994187 Ki = 88 nM T27812 CW0B4J 11034392 Ki = 1990 nM T27812 CEK01S 11044358 IC50 > 100000 nM T27812 CZ35QF 11045269 Ki = 1030 nM T27812 CY39BP 11046378 Ki = 15050 nM T27812 C2ZB0J 11059071 Ki = 1800 nM T27812 C3XW2P 11077246 Ki = 55.9 nM T27812 CIL61D 11077445 Ki = 2.3 nM T27812 C9KZ6L 11091998 Ki = 246 nM T27812 CFI32S 11095339 Ki > 10000 nM T27812 CXNV12 11102187 Ki = 41 nM T27812 C2IN5D 11102683 Ki = 160 nM T27812 CFMW85 11121384 Ki = 2810 nM T27812 C2ALP4 11130459 Ki = 38.1 nM T27812 CR6J8C 11130848 IC50 = 280 nM T27812 CLRV35 11134191 Ki = 45 nM T27812 C8W5NR 11145001 Ki = 85 nM T27812 C36VJK 11149970 Ki = 70.2 nM T27812 CT7Z9R 11150712 Ki = 14.8 nM T27812 C39INR 11150726 Ki = 199 nM T27812 CP7O3X 11161917 Ki = 80.9 nM T27812 CKB2H1 11163292 IC50 = 3600 nM T27812 CK27CU 11164446 Ki = 48.6 nM T27812 C1JC7S 11164569 IC50 = 104 nM T27812 C7OEX0 11174494 Ki = 4 nM T27812 CY67TG 11175450 IC50 = 862 nM T27812 CLE8G5 11176087 Ki = 0.171 nM T27812 C8KSG5 11177435 IC50 > 1000 nM T27812 CAN73X 11189693 IC50 > 3000 nM T27812 C1VIN4 11190988 Ki = 56 nM T27812 CHU5B0 11191321 Ki = 12 nM T27812 CM1T4L 11197267 IC50 = 2180 nM T27812 C01AFD 11200476 Ki = 16 nM T27812 CDMQ34 11202474 IC50 = 32.7 nM T27812 CPX23W 11209208 IC50 = 1960 nM T27812 CYQ65M 11214030 Ki = 5.7 nM T27812 C3VT2W 11219249 Ki > 10000 nM T27812 CVXM03 11221557 IC50 = 20 nM T27812 CCR0V5 11224454 Ki = 71.3 nM T27812 CV2R8E 11224953 Ki = 23 nM T27812 C3RO9W 11225779 Ki = 3.2 nM T27812 CA39QR 11227406 Ki = 2900 nM T27812 CR7IZ6 11231488 IC50 = 441 nM T27812 CG71SY 11233991 IC50 = 15 nM T27812 CQ7YK3 11244194 IC50 = 1525 nM T27812 CFC3D9 11246169 IC50 = 4.5 nM T27812 C6PUQ7 11246478 IC50 = 386 nM T27812 CQ0WO7 11248650 IC50 = 44.7 nM T27812 CPVA01 11255359 IC50 = 2600 nM T27812 CXNM72 11259744 Ki = 7.7 nM T27812 C5PWC6 11260018 Ki = 41 nM T27812 CPBA31 11260140 IC50 = 69.6 nM T27812 C8JW3Z 11260311 IC50 = 2.1 nM T27812 C6IRX4 11265803 Ki = 15.11 nM T27812 CG4R6Y 11266831 Ki > 100 nM T27812 C9S3BR 11267769 IC50 > 25000 nM T27812 C2JP5V 11270594 IC50 = 899 nM T27812 CZ8DY9 11271808 Ki = 3.5 nM T27812 C8YKS1 11271864 IC50 = 43.6 nM T27812 C6A0RY 11276613 Ki = 30 nM T27812 C27GXZ 11277680 Ki > 10000 nM T27812 CXH8G3 11278436 IC50 = 110 nM T27812 CW13FD 11280199 IC50 = 61.5 nM T27812 CC03FY 11287716 IC50 = 170 nM T27812 CH4EN9 11293572 IC50 = 25.2 nM T27812 C4U7GJ 11293591 IC50 = 1026 nM T27812 CG9TM7 11293593 Ki = 179.3 nM T27812 C57GTA 11299968 IC50 = 2430 nM T27812 CP26RV 11300496 Ki = 19 nM T27812 C3F7NY 11301501 IC50 = 7 nM T27812 CKQ7E8 11301538 Ki = 92.26 nM T27812 CV1LG4 11301893 IC50 = 21 nM T27812 CG0A3L 11303781 IC50 = 24.6 nM T27812 C7VS0M 11306100 Ki = 4.5 nM T27812 CS3BL0 11310988 Ki = 0.18 nM T27812 CUXZ91 11311148 IC50 = 1070 nM T27812 C2GZD3 11311204 Ki > 10000 nM T27812 C2S0GP 11313610 IC50 = 154 nM T27812 CM67PT 11318438 Ki = 13 nM T27812 CCJA60 11323414 Ki = 13 nM T27812 CKUG30 11327798 IC50 = 24.1 nM T27812 CCF56T 11334373 IC50 = 40 nM T27812 CBA4U5 11335494 IC50 = 440 nM T27812 CVL65D 11335835 IC50 = 3200 nM T27812 CF2X6Y 11336016 Ki = 3 nM T27812 CP6VZ2 11339973 IC50 = 300 nM T27812 CH83FN 11346324 Ki = 2.04 nM T27812 CXZ82E 11347860 IC50 = 2669 nM T27812 C3O0EP 11349976 IC50 = 6102 nM T27812 C1EGH7 11350339 IC50 = 42.6 nM T27812 C4ZP2J 11358065 IC50 > 9500 nM T27812 C8J5NW 11361155 IC50 = 8700 nM T27812 CR5S4A 11368527 Ki > 10000 nM T27812 C6A9TH 11373342 IC50 = 442 nM T27812 CV5XE3 11373704 IC50 = 128 nM T27812 C2N6CR 11374428 IC50 = 82.4 nM T27812 CS9D3C 11374767 IC50 = 27.9 nM T27812 CWV4P8 11375860 IC50 = 144 nM T27812 C6HFW9 11382841 IC50 = 20.5 nM T27812 CHQ9V1 11383270 Ki = 25.3 nM T27812 C3IJD5 11385494 IC50 = 1860 nM T27812 C4JVS8 11385652 Ki = 2.6 nM T27812 C7MN8V 11391287 IC50 = 2040 nM T27812 C7XOK1 11394095 IC50 = 42.2 nM T27812 C6CAV8 11394411 IC50 = 20 nM T27812 CE85CL 11415039 IC50 = 2350 nM T27812 CE5C4L 11418868 IC50 > 1000 nM T27812 CE2TS1 11425104 Ki > 10000 nM T27812 CCD2G1 11426012 IC50 = 17 nM T27812 CU4H7W 11426687 Ki = 518 nM T27812 CRH2D8 11428089 IC50 = 24.4 nM T27812 CGYC26 11442723 IC50 = 218 nM T27812 C2R6EU 11447499 Ki = 2 nM T27812 C6E3VO 11449834 Ki = 2460 nM T27812 CMH9J5 11450298 IC50 = 10 nM T27812 CX3ZU0 11450539 IC50 = 400 nM T27812 CNS8J9 11459667 Ki > 10000 nM T27812 CZAV70 11463320 IC50 = 1214 nM T27812 CT73UV 11463955 IC50 = 400 nM T27812 CF5R1Z 11463970 IC50 = 2000 nM T27812 C9L2AH 11474847 IC50 > 100000 nM T27812 CZ5SF1 11477432 IC50 = 70.6 nM T27812 C2X3OY 11483535 Ki = 1.83 nM T27812 C3QOL9 11484260 IC50 = 249 nM T27812 CK54EC 11485068 IC50 = 84.7 nM T27812 CC7O5G 11485868 IC50 = 64 nM T27812 CZ7X9M 11492164 IC50 = 2721 nM T27812 C7G5HP 11492305 Ki = 6885 nM T27812 CA8KE0 11492902 IC50 = 4.5 nM T27812 C3XD4T 11493035 IC50 = 1540 nM T27812 C2NJY3 11499666 IC50 = 111 nM T27812 C2X7HI 11499753 Ki > 10000 nM T27812 C7UJM8 11499957 IC50 = 540 nM T27812 CDC5I4 11499958 IC50 = 870 nM T27812 CXR70Z 11500795 Ki = 1650 nM T27812 CIN4B7 11500848 IC50 = 17 nM T27812 C3B0LO 11501191 Ki = 151 nM T27812 C1RQO0 11503600 Ki = 14 nM T27812 CR1K9A 11504964 Ki = 30 nM T27812 C2Y0JA 11505593 Ki = 68 nM T27812 CS1YI5 11506975 IC50 = 2576 nM T27812 C9OV2L 11507416 IC50 = 130 nM T27812 CZ61OG 11509486 Ki = 6.5 nM T27812 CNAW60 11511082 IC50 = 2 nM T27812 C6FA1G 11513575 Ki = 94 nM T27812 CM3P5D 11514441 Ki = 4100 nM T27812 C4DB0Z 11515426 IC50 = 33 nM T27812 C5MSI4 11517190 Ki = 4.3 nM T27812 CG51XI 11518064 Ki = 107 nM T27812 CSM9N1 11518191 IC50 = 530 nM T27812 C9XYF3 11521964 Ki > 10000 nM T27812 C3E1RM 11528759 Ki = 10 nM T27812 CFL1A3 11528838 Ki = 17 nM T27812 C75FPD 11529874 IC50 > 400 nM T27812 C3IBX7 11529992 IC50 = 93 nM T27812 C38QFE 11530118 Ki = 959 nM T27812 CWM49N 11535974 Ki = 59 nM T27812 C6SCW7 11536158 Ki = 21 nM T27812 CDM6F9 11536862 Ki = 2680 nM T27812 CE7KD1 11539564 IC50 = 26 nM T27812 CI4RN5 11539608 Ki = 5.7 nM T27812 C32SDT 11540601 Ki = 19 nM T27812 CC67XR 11543737 IC50 = 2.4 nM T27812 CGV24I 11544186 IC50 = 5 nM T27812 C0AP8I 11546190 IC50 = 4.7 nM T27812 CQ53AN 11546625 Ki = 42 nM T27812 CUQ3H4 11546759 IC50 = 150 nM T27812 C8VB1F 11547090 IC50 = 170 nM T27812 CQ74AN 11547594 IC50 > 1000 nM T27812 CWCU85 11548538 Ki = 41 nM T27812 CTXP63 11550888 IC50 = 35 nM T27812 C9VC7O 11551780 IC50 = 1780 nM T27812 C51PVS 11558708 IC50 = 72 nM T27812 C3RMI1 11559300 Ki = 1610 nM T27812 CJ1YS8 11561036 IC50 = 26 nM T27812 CY71DQ 11562044 Ki = 13 nM T27812 CH9MP0 11566229 Ki = 415 nM T27812 C1VF0P 11566266 Ki = 160 nM T27812 CDP9Z0 11566316 Ki = 179 nM T27812 C8C1VW 11566318 Ki = 36 nM T27812 CIE3O7 11566487 Ki = 630 nM T27812 CJAE31 11572186 Ki = 41 nM T27812 CZD62R 11572546 IC50 = 5.2 nM T27812 CCWG81 11573514 Ki = 143 nM T27812 CMX60P 11573849 IC50 = 5 nM T27812 C6JC2T 11580039 Ki > 10000 nM T27812 CD5XT0 11580456 IC50 = 38 nM T27812 CZ1QI8 11582342 Ki = 2.7 nM T27812 C2J9NU 11582508 Ki = 5.3 nM T27812 C2T6RF 11584839 Ki = 53 nM T27812 CZ2L0H 11586759 Ki = 5.7 nM T27812 CMZ54K 11587069 Ki = 2.1 nM T27812 C3LAI9 11587242 IC50 = 32 nM T27812 CY3A4K 11587772 Ki = 16 nM T27812 CU8F6B 11588595 IC50 = 38 nM T27812 C5Q1VL 11590382 Ki = 12 nM T27812 CI12ZR 11592176 Ki = 127 nM T27812 CTX5I8 11593896 Ki = 7.4 nM T27812 CW1CO6 11594137 IC50 = 130 nM T27812 CZ6US0 11594677 IC50 = 3300 nM T27812 CJ27XH 11594827 Ki = 9.69 nM T27812 C46AUZ 11597035 Ki = 3.2 nM T27812 CAD20M 11598831 Ki = 450 nM T27812 C9YR3G 11599258 Ki = 136 nM T27812 C7UFA1 11600778 IC50 > 10000 nM T27812 C6YB7K 11602095 Ki = 133 nM T27812 C5R2TD 11608403 Ki = 0.58 nM T27812 CE4GZ0 11609767 Ki = 5080 nM T27812 C6HLN8 11610150 Ki = 68 nM T27812 CN78BY 11612528 IC50 > 1000 nM T27812 C5PZF3 11615635 Ki = 8.9 nM T27812 C8JAM4 11616357 IC50 = 1 nM T27812 CCM6U9 11616771 Ki = 730 nM T27812 C1F4DL 11618807 Ki = 2 nM T27812 CI63EU 11619202 IC50 = 53 nM T27812 CUQ63N 11620342 Ki = 8.8 nM T27812 CI2VM7 11620991 Ki = 22 nM T27812 C5FQR2 11622909 Ki = 6.5 nM T27812 C32TIR 11623136 Ki = 1.8 nM T27812 C4YI2U 11623560 IC50 = 161 nM T27812 C1KD4Z 11623823 IC50 = 13 nM T27812 C86SZO 11624458 IC50 = 44 nM T27812 CYEH35 11627756 Ki = 286 nM T27812 C0I1YV 11628203 Ki = 58 nM T27812 CU61OB 11630020 Ki = 38 nM T27812 CA8IM9 11630375 Ki = 5900 nM T27812 CF0QR8 11630988 Ki = 6 nM T27812 CE8PC0 11632364 Ki = 4 nM T27812 CEZJ35 11633082 IC50 = 350 nM T27812 CK4M2L 11633374 Ki = 8.2 nM T27812 CQX2N5 11634999 IC50 = 570 nM T27812 CXJ73O 11638552 Ki = 28 nM T27812 CQ1U9W 11638962 Ki = 266 nM T27812 CU9AE6 11641636 IC50 > 1000 nM T27812 CGD21T 11642147 IC50 = 91 nM T27812 CGA8P4 11644537 Ki = 6.5 nM T27812 C3VOG6 11644931 IC50 = 14.5 nM T27812 CA9QZ5 11647367 Ki = 11 nM T27812 C8T9RB 11647974 IC50 = 57 nM T27812 C7XZ9J 11648391 Ki = 15 nM T27812 C97OLY 11649733 Ki = 82 nM T27812 CX2ZD7 11650267 IC50 = 127 nM T27812 C7BM5S 11650367 Ki = 76 nM T27812 C3OC6J 11650990 Ki = 1490 nM T27812 CZV1D5 11653516 Ki = 4.8 nM T27812 C1HDM5 11653679 Ki = 56.6 nM T27812 CM2E6F 11654898 IC50 = 2.9 nM T27812 CX7FR8 11655728 Ki = 28.84 nM T27812 CL4AJ0 11658719 IC50 = 4041 nM T27812 CWO6X9 11658763 Ki = 230 nM T27812 CAZN26 11659436 IC50 = 25 nM T27812 CF92SM 11659664 Ki = 9 nM T27812 C0KH7D 11660186 IC50 = 27 nM T27812 CN7J5K 11661512 Ki = 3.8 nM T27812 C50QHI 11661655 IC50 = 210 nM T27812 CIX54K 11666319 IC50 = 96 nM T27812 C1SYE2 11667017 IC50 = 41 nM T27812 C5WB3G 11668368 Ki = 2 nM T27812 CG1Q3H 11668849 Ki = 24 nM T27812 CKT39R 11669791 Ki = 135 nM T27812 CJ9Z8D 11671232 Ki = 100 nM T27812 C98NXK 11671382 Ki = 38 nM T27812 CEZ12X 11673089 Ki = 100 nM T27812 CT3BP5 11674529 Ki = 39 nM T27812 C79PHA 11678447 Ki = 43 nM T27812 C5Q3ZU 11680542 Ki = 15.85 nM T27812 CZHQ32 11683136 IC50 = 130 nM T27812 C2DBG7 11687579 IC50 = 31 nM T27812 C0Y6OR 11687843 Ki = 124 nM T27812 CL20PI 11690524 Ki = 6.5 nM T27812 CZ8TN6 11690910 Ki = 4.3 nM T27812 C3F9LC 11690966 Ki = 21 nM T27812 CD2I0Y 11694324 Ki = 0.68 nM T27812 C8R7TP 11694495 IC50 = 30 nM T27812 C6T8ZD 11694789 IC50 = 68 nM T27812 CU4D2Q 11701406 Ki = 14 nM T27812 CL19UR 11701869 IC50 = 40 nM T27812 CYN4H9 11702602 Ki > 100 nM T27812 CJ20GB 11705241 IC50 > 1000 nM T27812 CJ53MI 11705830 IC50 > 1000 nM T27812 C5OZD6 11706276 Ki = 280 nM T27812 CZB5P9 11709831 Ki = 229 nM T27812 C4M9AU 11710505 Ki = 222 nM T27812 CHK5I2 11712756 Ki = 31.62 nM T27812 CQWL60 11713341 Ki = 230 nM T27812 C18ZHK 11713731 Ki = 16 nM T27812 CHRM03 11716290 IC50 = 791 nM T27812 CKQ03I 11716308 IC50 = 225 nM T27812 CN2L4J 11716660 IC50 = 1.7 nM T27812 CX9VH0 11720815 Ki = 50.12 nM T27812 C6I5HN 11722722 IC50 = 9.6 nM T27812 C9BD4J 11723014 Ki = 170 nM T27812 CL7OG6 11739995 IC50 = 73 nM T27812 C4MC2V 11740717 Ki = 0.01 nM T27812 C6IQ8O 11751072 IC50 = 217 nM T27812 CB8A6W 11762106 IC50 = 6 nM T27812 C2QZI5 11771101 Ki = 50.58 nM T27812 C2M8JW 11777763 IC50 = 18 nM T27812 CMX8Z2 11778484 IC50 = 200 nM T27812 CN4Y8B 11778700 IC50 = 41 nM T27812 CX7TO1 11785068 Ki = 26 nM T27812 CE4Q9W 11785961 Ki = 17 nM T27812 CKNE31 11791987 Ki > 10000 nM T27812 CW15BI 11794260 Ki = 300 nM T27812 CQGL96 11797680 Ki = 47 nM T27812 CJO0Q6 11818515 Ki = 2177 nM T27812 C9ZQ4F 11826809 Ki = 370 nM T27812 C0ZR7C 11845636 IC50 = 732 nM T27812 CDTQ46 11845643 IC50 = 116 nM T27812 CJ9D3N 11845645 IC50 = 42.7 nM T27812 CO81MR 11845815 IC50 = 181 nM T27812 CJ4TH0 11845817 IC50 = 53.5 nM T27812 CVOC94 11845819 IC50 = 59.7 nM T27812 C3L4QY 11845822 IC50 = 18.7 nM T27812 CL0OH3 11845824 IC50 = 17.4 nM T27812 CU39AH 11846005 IC50 = 883 nM T27812 C58BSD 11846181 IC50 = 197 nM T27812 CNVY54 11846183 IC50 = 37.3 nM T27812 C7P8FK 11846185 IC50 = 59.9 nM T27812 CX1B6K 11846187 IC50 = 36.3 nM T27812 C2UT9D 11846746 IC50 = 6 nM T27812 CRX17H 11855337 Ki = 1.1 nM T27812 CXLW54 11948707 Ki > 10000 nM T27812 C8EJ6H 11949672 IC50 = 1400 nM T27812 CK13QD 11953409 Ki = 29000 nM T27812 C8JQL7 11957735 IC50 > 10000 nM T27812 C5QB3M 11963972 IC50 = 700 nM T27812 CAW2Y1 12000105 Ki = 296 nM T27812 C3LG9X 12017337 Ki = 220 nM T27812 CX2TQ7 12111555 IC50 = 260 nM T27812 C49HJG 12122109 Ki = 185 nM T27812 CUFP52 12149037 IC50 = 927 nM T27812 CT4RA6 12204576 Ki = 39 nM T27812 CK6WG1 12276477 IC50 = 1517 nM T27812 C4S0VH 12371032 EC50 = 29600 nM T27812 C93RWQ 12371034 IC50 = 300 nM T27812 C2MP5H 12559279 IC50 > 10000 nM T27812 CV70JI 12634880 Ki = 36 nM T27812 C6MH2K 12646716 IC50 = 35400 nM T27812 CG3F5T 12674078 IC50 = 220 nM T27812 CQV9X3 12674079 IC50 > 1000 nM T27812 C1OPN4 12674080 IC50 > 1000 nM T27812 CE9L3N 12674083 IC50 > 1000 nM T27812 C9WU7D 12674084 IC50 > 1000 nM T27812 C50WCY 12674086 IC50 = 60 nM T27812 C5UY6P 12674087 IC50 > 1000 nM T27812 C2ZE8Y 12674088 IC50 > 1000 nM T27812 C0KR1M 12884652 Ki = 800 nM T27812 C3B8LI 12968865 Ki = 66.4 nM T27812 CB8V2N 12968873 Ki = 38.9 nM T27812 C72BFQ 12968875 Ki = 42.6 nM T27812 C8C5KI 12968876 Ki = 62.4 nM T27812 C13WPY 12968877 Ki = 46.2 nM T27812 CE5Y2W 12980713 IC50 = 1.63 nM T27812 CM78FI 12999584 IC50 = 99 nM T27812 CCG14E 13091356 Ki = 255 nM T27812 CYN95Z 13091359 Ki = 316 nM T27812 C2WY8Z 13361400 Ki > 7000 nM T27812 C9CF3W 13520310 IC50 = 123 nM T27812 C1FAP2 13520317 IC50 = 88 nM T27812 CQV86I 13718739 IC50 > 10000 nM T27812 CGY6Q3 13718746 IC50 > 10000 nM T27812 C0KU4R 13718753 IC50 = 3100 nM T27812 C12NSL 13718761 IC50 = 5400 nM T27812 CI6TP9 13903189 Ki = 0.9 nM T27812 CHJ27K 13903191 Ki = 0.27 nM T27812 C4KU1J 14014888 IC50 > 10000 nM T27812 CQI9F6 14571114 Ki = 2050 nM T27812 C9GEN5 14674210 IC50 > 10000 nM T27812 C57QFI 14930273 IC50 = 0.36 nM T27812 C4L7WJ 14973208 IC50 = 210 nM T27812 C4GY9E 14973209 IC50 = 160 nM T27812 C3KM9T 14973210 IC50 = 910 nM T27812 CB3W8C 14973216 IC50 = 19 nM T27812 C8UBJ4 15015316 Ki = 6.4 nM T27812 CJ8WL9 15015330 Ki = 0.7 nM T27812 CO5C4K 15029820 IC50 = 160 nM T27812 C0P5LY 15069893 Ki = 4.3 nM T27812 CE4T7Z 15069894 Ki = 21 nM T27812 C8SXL1 15069905 Ki = 0.96 nM T27812 CMI6C8 15113388 Ki = 1450 nM T27812 C27ZJA 15113390 Ki = 1570 nM T27812 CD24IR 15115364 IC50 = 250 nM T27812 CDC3Q9 15132120 IC50 = 20 nM T27812 CTZ61G 15132121 IC50 = 12 nM T27812 C2T1UK 15290836 IC50 = 0.34 nM T27812 CO6P8K 15405849 Ki = 7.77 nM T27812 CZ01RO 15547884 Ki = 50 nM T27812 CYQ2L9 15547887 Ki = 36 nM T27812 CMP83C 15550585 IC50 = 33 nM T27812 C53JMI 15639786 Ki = 4 nM T27812 C1FLJ0 15639787 Ki = 4.2 nM T27812 C4OT1S 15639792 Ki = 6 nM T27812 CW8M6S 15952123 IC50 = 5500 nM T27812 CT12KQ 15980807 Ki = 184 nM T27812 C5HQT6 15980808 Ki = 26 nM T27812 C4JT9L 15980809 Ki = 28 nM T27812 C76PIS 15980810 Ki = 8 nM T27812 CF4Z2U 15980852 Ki = 340 nM T27812 CZ39MX 15980853 Ki = 27 nM T27812 C0H7GI 15980854 Ki = 112 nM T27812 CTH2S5 15980895 Ki = 15 nM T27812 C58TFK 15981911 Ki = 93 nM T27812 C6T5GH 15981916 Ki = 106 nM T27812 CJ7TI6 15981917 Ki = 37 nM T27812 CTU6F4 15982036 Ki = 62 nM T27812 CFPV59 15982037 Ki = 31 nM T27812 CIX70J 15982171 Ki = 4767 nM T27812 CM6O3G 15983286 IC50 = 105 nM T27812 CRN92T 15983453 Ki = 1137 nM T27812 CYO4G3 15983454 Ki = 768 nM T27812 CMD02L 15983456 Ki = 2333 nM T27812 C4SJF0 15983457 Ki = 2000 nM T27812 CP94BW 15983458 Ki = 147 nM T27812 CM12TW 15983459 Ki = 12 nM T27812 C7X0TJ 15983575 Ki = 189 nM T27812 CP96DT 15983576 Ki = 70 nM T27812 CWQ59P 15983578 Ki = 302 nM T27812 CLV05C 15983579 Ki = 32 nM T27812 CF1H7C 15983580 Ki = 120 nM T27812 CY5U3T 15983703 Ki = 362 nM T27812 CEG95K 15983705 Ki = 226 nM T27812 CX2L9Q 15983706 Ki = 26 nM T27812 CDJ9B2 15983708 Ki = 141 nM T27812 C08HXO 15983836 Ki = 1333 nM T27812 C8P2AR 15983838 Ki = 826 nM T27812 CE9Z5F 15983840 Ki = 66 nM T27812 C9K2MU 15983841 Ki = 26 nM T27812 C3BLG0 16005416 Ki = 2.5 nM T27812 CA91OD 16005497 Ki = 16.7 nM T27812 C8V1IK 16005500 Ki = 88 nM T27812 CO0E2Y 16006089 Ki = 3.3 nM T27812 CDB1W5 16006612 Ki = 1.3 nM T27812 CQV08D 16006719 Ki = 66 nM T27812 C89XFJ 16007138 Ki = 50 nM T27812 CG60DM 16038376 IC50 > 3000 nM T27812 C37FIP 16047544 Ki = 2716 nM T27812 CL0B8J 16063251 IC50 = 14 nM T27812 C4FG6R 16066745 EC50 = 3981.07 nM T27812 C30UFT 16066811 IC50 = 1680 nM T27812 CO58NM 16067544 IC50 = 1750 nM T27812 C4LFH6 16067545 IC50 = 1150 nM T27812 C5KHE3 16067546 IC50 > 3000 nM T27812 CR8F9E 16067547 IC50 = 2550 nM T27812 CE4A2K 16067549 IC50 = 1950 nM T27812 CJRU09 16067550 IC50 = 1350 nM T27812 C8PL4S 16067551 IC50 > 3000 nM T27812 CTS91K 16067641 IC50 = 4311 nM T27812 CP54FR 16067643 IC50 = 4565 nM T27812 CPLR62 16067646 IC50 = 166 nM T27812 C0VK4Y 16067647 IC50 = 3100 nM T27812 CQ4P2J 16067648 IC50 = 273 nM T27812 CAY61X 16067730 IC50 = 2995 nM T27812 C3QMW5 16067734 IC50 = 1910 nM T27812 CLY3X5 16067834 IC50 = 1408 nM T27812 C8I6EM 16067835 IC50 = 1208 nM T27812 C83KQX 16067839 IC50 > 3000 nM T27812 CJ24NE 16067840 IC50 = 330 nM T27812 C2RA5B 16067943 IC50 = 290 nM T27812 CTG78M 16067944 IC50 = 483 nM T27812 CEVD42 16091071 Ki = 608 nM T27812 C7UOM4 16092107 Ki = 8 nM T27812 CH74RZ 16102752 IC50 = 3300 nM T27812 C6OR3H 16102755 Ki = 5000 nM T27812 C9SH0B 16102756 IC50 = 1800 nM T27812 CA75KZ 16102757 Ki = 2900 nM T27812 C1L9HQ 16102758 Ki = 900 nM T27812 CMUI02 16102759 Ki = 1100 nM T27812 CLO54U 16102760 IC50 = 210 nM T27812 C3SEF2 16102761 Ki = 700 nM T27812 CYF03S 16102762 Ki = 3900 nM T27812 C4N9BG 16102763 IC50 = 4200 nM T27812 C2HLF8 16102765 IC50 = 550 nM T27812 CTX94E 16102766 Ki = 450 nM T27812 C9HLB7 16102767 Ki = 950 nM T27812 CLHY18 16102768 IC50 = 2600 nM T27812 CG90ID 16102769 Ki = 1700 nM T27812 CH53XS 16102770 Ki = 1300 nM T27812 CQS4V1 16112801 IC50 > 10000 nM T27812 CJ32XS 16113210 IC50 = 13 nM T27812 C9UYE0 16126667 Ki = 572 nM T27812 C4QCP3 16494915 IC50 > 10 nM T27812 C2VQS3 16640939 IC50 = 28 nM T27812 C6P4BX 16656803 IC50 = 79 nM T27812 CZ2IS9 16660294 Ki > 10000 nM T27812 CW40DA 16678084 IC50 = 452 nM T27812 CH4Y2D 16681434 IC50 = 100 nM T27812 CB7G3R 16718920 IC50 > 10000 nM T27812 CDT5V8 16721129 Ki = 3.8 nM T27812 C3J9ZX 16730430 IC50 = 8.9 nM T27812 CL5G7A 16730754 Ki = 440 nM T27812 CUG5B8 16747689 Ki = 0.72 nM T27812 C50YME 16747877 Ki = 2390 nM T27812 CY8QO6 16748004 Ki = 5700 nM T27812 CY2FL4 16748005 Ki = 1820 nM T27812 C9CQ1B 16748006 Ki = 5200 nM T27812 COGJ31 16748007 IC50 = 1840 nM T27812 CPF2K0 16748165 Ki = 580 nM T27812 CM1L6Q 16748381 Ki = 3590 nM T27812 CG5FU0 16748382 Ki = 1720 nM T27812 CYN9W8 16748383 Ki = 1640 nM T27812 CM89SX 16748512 Ki = 3670 nM T27812 C1ZQX9 16748513 Ki = 7710 nM T27812 CM46NI 16748623 Ki = 740 nM T27812 C9W7LH 16748731 Ki = 870 nM T27812 CJ9S7I 16748848 Ki = 653 nM T27812 CXH10U 16748849 Ki = 1500 nM T27812 C37DZJ 16748949 Ki = 2710 nM T27812 CTJ2Z3 16748950 IC50 = 377 nM T27812 C1L8DV 16748951 Ki = 2940 nM T27812 CQV8E0 16783706 IC50 > 400 nM T27812 CN4HB8 18391094 Ki = 1900 nM T27812 CH39LP 18391096 Ki = 3700 nM T27812 CMIO28 18428690 IC50 = 12 nM T27812 CT0I8X 18428716 Ki = 1.7 nM T27812 CUEV14 18446803 IC50 > 6000 nM T27812 C03IZO 18623856 IC50 = 5.87 nM T27812 CJ6ZF2 18756309 IC50 = 2580 nM T27812 C9JD5Y 19360456 IC50 = 21 nM T27812 CYFJ81 19926671 IC50 = 1.68 nM T27812 C21LXU 20055336 Ki = 4 nM T27812 C8ICF9 20111627 IC50 < 1 nM T27812 CQ6PB2 20443021 Ki = 150 nM T27812 CPVF37 20443023 Ki = 250 nM T27812 CX9HZ2 20443040 Ki = 88 nM T27812 CC2G4J 20611340 IC50 = 5.95 nM T27812 C6R8AM 20631904 Ki = 2.1 nM T27812 C81FRQ 20636465 Ki = 19 nM T27812 CXQM78 20695745 IC50 > 100 nM T27812 CEO8W1 21116177 IC50 > 10000 nM T27812 C7Y0HC 21302486 Ki = 31 nM T27812 C2EO0C 21302505 Ki = 27 nM T27812 CRV56X 21365270 IC50 = 102 nM T27812 C3T5HF 21509921 Ki = 2187.76 nM T27812 CFN81Q 21527771 Ki = 2228 nM T27812 CH59WN 21533446 Ki = 160 nM T27812 C27GSH 21539381 IC50 = 99.2 nM T27812 C1MR4F 21959106 IC50 = 2.19 nM T27812 C42AIN 21959117 IC50 = 7990 nM T27812 C0AW7O 21959124 IC50 = 1.24 nM T27812 C0OIX1 22019270 IC50 = 4.99 nM T27812 CXQK98 22197529 Ki > 10000 nM T27812 C2X0TW 22337167 IC50 > 100000 nM T27812 CR4T9J 22337182 Ki > 100000 nM T27812 CQUY92 22386812 Ki = 2850 nM T27812 C7O8WZ 22386894 Ki = 10.3 nM T27812 CMDI47 22386922 Ki = 4224 nM T27812 CW5M2S 22419110 Ki = 9.63 nM T27812 CPI8Q3 22419116 IC50 = 20.4 nM T27812 CU8YV6 22468266 Ki = 4.9 nM T27812 CF6P4V 22468271 Ki = 52 nM T27812 CXKF39 22638783 IC50 = 25 nM T27812 C49VCE 22675297 Ki = 37.5 nM T27812 CIC7F6 22675312 Ki = 13.9 nM T27812 CBCK13 22675339 Ki = 51.2 nM T27812 CPU6C8 22675347 Ki = 37.6 nM T27812 C85YGH 22675350 Ki = 25.6 nM T27812 CP41JS 22675387 Ki = 12.4 nM T27812 C5R7JT 22675398 Ki = 18.7 nM T27812 CV2XH0 22798952 IC50 = 724.44 nM T27812 CD63RO 22860156 IC50 = 1830 nM T27812 CPH6L4 22966050 Ki = 50 nM T27812 CAP1B3 23001840 IC50 = 60 nM T27812 CYPV48 23378645 IC50 = 12 nM T27812 C4ATJ7 23378652 IC50 = 2 nM T27812 CUF6W8 23378663 IC50 = 6 nM T27812 C57EFO 23378743 IC50 = 7 nM T27812 C98KLS 23378746 IC50 = 5 nM T27812 C2QXK6 23449967 IC50 = 4800 nM T27812 CUD3Y7 23449968 IC50 = 4.67 nM T27812 CMEV08 23449969 IC50 > 10000 nM T27812 C9QD6T 23449971 IC50 = 180 nM T27812 CCP24F 23449972 IC50 = 35400 nM T27812 C31ASG 23449975 IC50 = 30 nM T27812 C2HK1Z 23449980 IC50 = 12 nM T27812 CP1A4B 23449981 IC50 > 30000 nM T27812 CW0D5K 23449986 IC50 = 107 nM T27812 CH8O4R 23449987 IC50 > 10000 nM T27812 CG08BF 23449988 IC50 > 60000 nM T27812 CHD8T7 23449989 IC50 > 50000 nM T27812 CL45FG 23519626 IC50 = 110 nM T27812 CDJR16 23519628 IC50 = 181 nM T27812 CF3SU0 23519629 IC50 = 25 nM T27812 C7YFT3 23582127 Ki = 6 nM T27812 C57MTL 23625757 Ki = 0.9 nM T27812 C6IF2N 23661687 Ki > 1000000 nM T27812 CNU2X4 23725134 IC50 > 1000 nM T27812 CSB9E8 24103136 IC50 = 22 nM T27812 C6ZE3Y 24180451 Ki = 2.3 nM T27812 C0I5RA 24180665 IC50 = 83 nM T27812 CFM03J 24208815 IC50 = 381 nM T27812 C60JDQ 24257988 IC50 = 1900 nM T27812 C56SPY 24258016 IC50 = 1600 nM T27812 CQ0KU9 24738459 Ki = 26 nM T27812 C91IVZ 24742317 IC50 = 14 nM T27812 C32IVO 24742475 IC50 = 320 nM T27812 CWGH86 24743352 IC50 = 13 nM T27812 CYBG40 24743354 IC50 = 420 nM T27812 CG3XD5 24743436 IC50 = 26 nM T27812 C61QPT 24748794 Ki = 1.1 nM T27812 C9P2NE 24748795 Ki = 1.3 nM T27812 CYRZ48 24749837 Ki = 0.1 nM T27812 C4Y0BF 24749952 Ki = 0.95 nM T27812 CJ2N8B 24749953 Ki = 5 nM T27812 CV30EH 24749955 Ki = 1.2 nM T27812 CPD4M8 24749956 Ki = 0.21 nM T27812 CO7TD4 24750311 Ki = 0.25 nM T27812 C4R9YO 24750312 Ki = 0.03 nM T27812 C60SIH 24750313 Ki = 0.05 nM T27812 C2ZJ3Q 24750421 Ki = 1.4 nM T27812 CV1K6O 24750422 Ki = 0.15 nM T27812 CQ1G3S 24750423 Ki = 17 nM T27812 C6GBU8 24762221 Ki = 50.12 nM T27812 C16YHA 24764464 IC50 = 112 nM T27812 CHI83W 24769038 IC50 = 0.023 nM T27812 C5ASY1 24773552 Ki = 0.29 nM T27812 C1FIS5 24773804 Ki = 1.26 nM T27812 C9KXC8 24773805 Ki = 0.31 nM T27812 CP1F6M 24782241 Ki = 12.59 nM T27812 CZ2XE7 24782243 Ki = 7.943 nM T27812 CJQ2X4 24782485 Ki = 15.85 nM T27812 CI7S2G 24782486 Ki = 1.259 nM T27812 CK5TO1 24782487 Ki = 63.1 nM T27812 CZ34RN 24782489 Ki = 15.85 nM T27812 CL5GS1 24786064 Ki = 7.943 nM T27812 CDQ58K 24799187 IC50 = 4 nM T27812 CTQ59S 24799364 IC50 = 15 nM T27812 C8LJY2 24799365 IC50 = 4.8 nM T27812 CO32ND 24799366 IC50 = 7.3 nM T27812 C6X0JS 24799545 IC50 = 3.9 nM T27812 CG24KB 24799546 IC50 = 140 nM T27812 C1QL3V 24799711 IC50 = 2.8 nM T27812 CH0Y9J 24800231 IC50 = 2.1 nM T27812 C10YFG 24800398 IC50 = 6.8 nM T27812 C3FYB5 24800577 IC50 = 94 nM T27812 C17RDK 24800578 IC50 = 58 nM T27812 C30UAB 24800743 IC50 = 7.3 nM T27812 C6SHG9 24800925 IC50 = 10 nM T27812 C0L6CF 24800927 IC50 = 7.4 nM T27812 CM2K4N 24801101 IC50 = 9 nM T27812 CP8T1L 24801102 IC50 = 6.6 nM T27812 CA8GT1 24801457 IC50 = 4.3 nM T27812 CW8GD6 24801458 IC50 = 6.6 nM T27812 CE25UP 24801459 IC50 = 4.3 nM T27812 CSK49W 24801626 IC50 = 6.3 nM T27812 C1NK4A 24801627 IC50 = 14 nM T27812 C9GK5S 24801792 IC50 = 88 nM T27812 CWH29M 24801795 IC50 = 2.4 nM T27812 C84TEM 24801797 IC50 = 3.3 nM T27812 CQN4W1 24802843 Ki = 7.943 nM T27812 C23ICW 24802846 Ki = 12.59 nM T27812 CX6ZB7 24802848 Ki = 12.59 nM T27812 CH30VR 24803009 Ki = 15.85 nM T27812 CH87VD 24803010 Ki = 1 nM T27812 CC78ZE 24803012 Ki = 7.943 nM T27812 C7C4UQ 24803014 Ki = 15.85 nM T27812 C17ISZ 24803180 Ki = 3.162 nM T27812 C4O8ZF 24803181 Ki = 15.85 nM T27812 C1W8NS 24803185 Ki = 1.585 nM T27812 C9LV3D 24803344 Ki = 6.31 nM T27812 C96CBA 24803345 Ki = 10 nM T27812 CJ4RO1 24804774 Ki = 25.12 nM T27812 CK84BF 24804775 Ki = 2.512 nM T27812 C1Z3OQ 24804941 Ki = 10 nM T27812 C6AE2U 24804942 Ki = 0.5012 nM T27812 C1ZYM4 24804943 Ki = 1 nM T27812 CN6UX3 24809704 Ki > 50000 nM T27812 C09QDS 24809705 Ki = 10000 nM T27812 C85LUK 24822173 IC50 = 5500 nM T27812 CPH72B 24825320 Ki = 88 nM T27812 C3LW5Z 24825321 Ki = 22 nM T27812 CHZS54 24825322 Ki = 220 nM T27812 C03LDP 24825323 Ki = 250 nM T27812 C2IB8H 24825324 Ki = 290 nM T27812 CQKH10 24825325 Ki = 540 nM T27812 CPN0C7 24825326 Ki = 190 nM T27812 CAV1B6 24825327 Ki = 1800 nM T27812 C0BR5C 24825328 Ki = 1800 nM T27812 CVQ8C7 24825329 Ki = 2500 nM T27812 CV72IA 24825330 Ki = 430 nM T27812 CL0DF1 24825331 Ki = 3300 nM T27812 CR2L5Q 24825332 Ki = 310 nM T27812 C9V6HW 24825333 Ki = 2000 nM T27812 CAD2R1 24825334 Ki = 1400 nM T27812 CR3FA2 24825335 Ki = 110 nM T27812 C17ZME 24825336 Ki = 190 nM T27812 C0M7CN 24825720 Ki = 51.29 nM T27812 CDC91N 24839550 Ki = 151.36 nM T27812 C6ZRA7 24849533 Ki = 12.59 nM T27812 C50XIV 24855884 Ki = 9 nM T27812 CJTY89 24855886 Ki = 17 nM T27812 C79FCO 24855918 Ki = 236 nM T27812 CJAC42 24855949 Ki = 229 nM T27812 C1SVD5 24855952 Ki = 12 nM T27812 CYQS46 24855953 Ki = 2.9 nM T27812 CGC54I 24855977 Ki = 14 nM T27812 CAF5W4 24855979 Ki = 36 nM T27812 C96KWD 24855980 Ki = 41 nM T27812 CEV3S9 24855981 Ki = 94 nM T27812 C3A6SC 24856010 Ki = 122 nM T27812 C5T6WF 24856012 Ki = 68 nM T27812 C2BG9R 24856014 Ki = 13 nM T27812 CS1VR8 24856015 Ki = 95 nM T27812 CG07AV 24856046 Ki = 702 nM T27812 C67OXE 24856047 Ki = 797 nM T27812 CW0J7T 24856048 Ki = 1400 nM T27812 CE2UI4 24856107 Ki = 5 nM T27812 C48LYD 24856108 Ki = 562 nM T27812 C0DUL3 24857666 IC50 = 46 nM T27812 CC8J1Z 24857667 IC50 = 1830 nM T27812 C9V5MT 24857668 IC50 = 84 nM T27812 C5QGY4 24857669 IC50 = 108 nM T27812 CSR8J4 24857759 IC50 = 1 nM T27812 C27EUV 24857839 IC50 = 26 nM T27812 CZ8TA6 24857854 IC50 = 25 nM T27812 C97SEP 24857858 Ki = 4.11 nM T27812 CBI5D7 24860769 IC50 = 110 nM T27812 C7COU6 24860831 IC50 = 660 nM T27812 CVO64M 24860832 IC50 = 1700 nM T27812 CL26KS 24860835 IC50 = 60 nM T27812 C7EHG5 24860898 IC50 = 855 nM T27812 C2X6VF 24860899 IC50 = 260 nM T27812 CAU07P 24860900 IC50 > 10000 nM T27812 CM9L7D 24860902 IC50 = 637 nM T27812 CZ3R7W 24860903 IC50 = 330 nM T27812 CG8T3J 24860904 IC50 = 540 nM T27812 CO51AG 24863961 Ki = 7105 nM T27812 CD9SF2 24863962 Ki = 9465 nM T27812 C3HK0J 24865725 Ki = 1584.89 nM T27812 C0O6FX 24865727 Ki = 398.11 nM T27812 CXD45U 24867041 IC50 = 12 nM T27812 CV1PY2 24878951 Ki = 3303 nM T27812 CK6JC4 24878953 Ki > 100000 nM T27812 C4SL0V 24879001 Ki > 100000 nM T27812 C3Z4JN 24879003 Ki > 10000 nM T27812 C56IDA 24879005 Ki = 3791 nM T27812 C23LNY 24879008 Ki > 100000 nM T27812 C9C8OH 24879010 Ki > 100000 nM T27812 C1ZRH6 24879054 Ki > 10000 nM T27812 CD17RE 24879056 Ki > 10000 nM T27812 CX20BZ 24879058 Ki > 10000 nM T27812 C9A2NF 24890939 Ki = 6.8 nM T27812 CG0Z8X 24893996 IC50 = 11 nM T27812 C46VNQ 24895014 IC50 = 405 nM T27812 CV9E4X 24895015 IC50 = 155 nM T27812 C8ER2O 24897032 IC50 = 196 nM T27812 C0Z4PW 24897264 IC50 = 183 nM T27812 C5HPS8 24897268 IC50 = 76 nM T27812 CT0HG9 24897269 IC50 = 2607 nM T27812 CB37QM 24897270 IC50 = 32 nM T27812 C7B3YH 24897482 IC50 = 73 nM T27812 CMP23U 24897483 IC50 = 286 nM T27812 CQ1N4S 24897484 IC50 = 41 nM T27812 CN3XK4 24897486 IC50 = 22 nM T27812 CH1PU0 24897487 IC50 = 17 nM T27812 CNH7C9 24897687 IC50 = 237 nM T27812 C48GLF 24897688 IC50 = 167 nM T27812 CTG6D4 24897689 IC50 = 55 nM T27812 C4FEQ6 24936132 Ki = 121 nM T27812 C61XEY 24937629 IC50 = 2983 nM T27812 C4G8UV 24937633 IC50 = 2042 nM T27812 C6I4YO 24937759 IC50 = 4589 nM T27812 C0BP8C 24939244 IC50 > 10000 nM T27812 C1GAD9 24946664 Ki = 16 nM T27812 CF26PB 24946667 Ki = 39 nM T27812 C9W1EB 24946668 Ki = 24 nM T27812 CWK21C 24947199 Ki = 14 nM T27812 CDI10X 24947200 Ki = 199 nM T27812 CO2TD9 24947376 Ki = 10 nM T27812 CIG62P 24947377 Ki = 159 nM T27812 CI6TP1 24947378 Ki = 16 nM T27812 CSL93K 24947379 Ki = 60 nM T27812 CY9X8Z 24947380 Ki = 16 nM T27812 C20BSY 24947381 Ki = 3 nM T27812 C3H5PJ 24947569 Ki = 5 nM T27812 CUM1C3 24947570 Ki = 46 nM T27812 CERD40 24947571 Ki = 9 nM T27812 CB2U7X 24947572 Ki = 8.7 nM T27812 CQ7Z6F 24947573 Ki = 11 nM T27812 CEGC24 24947574 Ki = 2.7 nM T27812 CSJ5I4 24947575 Ki = 4 nM T27812 C4Y7FP 24947750 Ki = 5.9 nM T27812 CA8VN2 24947751 Ki = 8.1 nM T27812 CYGT57 24947752 Ki = 28 nM T27812 CL60YE 24947753 Ki = 24 nM T27812 C1FSB7 24947760 Ki = 61 nM T27812 CFJ4O7 24947761 Ki = 29 nM T27812 CEW8C3 24947936 Ki = 155 nM T27812 CVZ7K9 24947937 Ki = 535 nM T27812 C72EWS 24947938 Ki = 363 nM T27812 C8TKG2 24947939 Ki = 37 nM T27812 C6BIR1 24947941 Ki = 11 nM T27812 C06TLI 24948121 Ki = 23 nM T27812 C2OK6I 24948317 Ki = 169 nM T27812 C9WPU6 24948318 Ki = 1480 nM T27812 C0BL9R 24948319 Ki = 245 nM T27812 C8MU7D 24948320 Ki = 42 nM T27812 CJ0M6T 24948507 Ki = 281 nM T27812 CW4X0E 24962988 Ki = 1110 nM T27812 C2XUP4 24963805 Ki = 1.8 nM T27812 C6DW3J 24964157 Ki = 0.7 nM T27812 CQ42YZ 24964158 Ki = 0.8 nM T27812 C4P5AD 24964159 Ki = 1.9 nM T27812 CP6SX7 24964160 Ki = 1.2 nM T27812 CP53AB 24964161 Ki = 30 nM T27812 C3YXJ9 24964162 Ki = 2.7 nM T27812 CZV16S 24964163 Ki = 24 nM T27812 C2PA7D 24964521 Ki = 13 nM T27812 CFPU09 24964522 Ki = 7.3 nM T27812 CYK2Q6 24964523 Ki = 3.5 nM T27812 CNU2L1 24964524 Ki = 12 nM T27812 C2L0PV 24964525 Ki = 1.4 nM T27812 C1X3LT 24964877 Ki = 5.9 nM T27812 CN7B3D 24964878 Ki = 1.3 nM T27812 C8KID6 24964879 Ki = 3.6 nM T27812 CB9C4E 24965063 Ki > 6000 nM T27812 CZXC58 24965064 Ki > 6000 nM T27812 CA3T8S 24965234 Ki = 1.2 nM T27812 COH49Y 24965236 Ki = 17 nM T27812 CK2I8F 24965237 Ki = 3.6 nM T27812 C9PVS1 24965238 Ki = 27 nM T27812 CY0IN2 24965589 Ki = 2 nM T27812 CL56YC 24965590 Ki = 1.4 nM T27812 C1SUL8 24965930 Ki = 3.4 nM T27812 CT39VO 24969452 IC50 = 300 nM T27812 CGZ60N 24969453 IC50 = 590 nM T27812 CKNQ63 25008443 IC50 = 5263 nM T27812 CZ6T5Q 25009937 Ki = 110 nM T27812 CQ9LS6 25022704 Ki = 823 nM T27812 C0HRL1 25024305 Ki = 6.31 nM T27812 C2RQX9 25024309 Ki = 7.943 nM T27812 C3W1NC 25024503 Ki = 79.43 nM T27812 CY0VU5 25025577 Ki = 25.7 nM T27812 CA20NZ 25025581 Ki = 0.1585 nM T27812 CU8A6N 25025776 Ki = 0.2512 nM T27812 C4I5LJ 25025778 Ki = 0.631 nM T27812 CPJD86 25025779 Ki = 0.07943 nM T27812 CN0U3C 25025780 Ki = 1.259 nM T27812 CFAZ02 25025782 Ki = 0.1995 nM T27812 CDX2C6 25025977 Ki = 0.1259 nM T27812 CRQ73B 25025978 Ki = 0.631 nM T27812 C9WQ5K 25025979 Ki = 0.2512 nM T27812 C16YGB 25029543 IC50 = 6000 nM T27812 CZX10T 25030029 IC50 = 2000 nM T27812 CZ7C0R 25030031 IC50 = 13300 nM T27812 CE89TZ 25030033 IC50 = 1500 nM T27812 CZOR47 25030035 IC50 = 110 nM T27812 CA4L5Q 25032786 IC50 > 1000 nM T27812 C6K4SH 25033519 IC50 = 4 nM T27812 CR5FX4 25059765 IC50 > 10000 nM T27812 CMVL70 25059766 IC50 > 1000 nM T27812 CED30A 25059770 IC50 > 1000 nM T27812 CJU9Y7 25060021 IC50 > 1000 nM T27812 C36PMH 25060023 IC50 > 1000 nM T27812 CHSB87 25060024 IC50 > 1000 nM T27812 CPT9X8 25066443 IC50 = 13 nM T27812 CPGZ03 25069239 Ki = 54.6 nM T27812 CT0R3H 25069240 Ki = 13.6 nM T27812 CX5JF4 25069241 Ki = 15.6 nM T27812 C1P4EC 25069242 Ki = 9.22 nM T27812 CCV27I 25069243 Ki = 30.8 nM T27812 C5BR0K 25069297 Ki = 110 nM T27812 CU34CX 25069298 Ki = 10.5 nM T27812 C0Z6YL 25069299 Ki = 9.1 nM T27812 C5Z9MA 25069300 Ki = 84.7 nM T27812 C1OGS2 25069301 Ki = 447 nM T27812 C53LJG 25069302 Ki = 160 nM T27812 CX74UK 25069353 Ki = 24.7 nM T27812 C8F6VC 25069354 Ki = 2520 nM T27812 C56RCY 25069355 Ki = 259 nM T27812 CI7SM5 25069356 Ki = 2720 nM T27812 CIWT97 25071015 Ki = 6.16 nM T27812 CP9J7Q 25071019 IC50 = 1700 nM T27812 C45AHR 25093400 IC50 = 8 nM T27812 C0DFW8 25093401 IC50 = 50 nM T27812 C67OHQ 25093402 IC50 = 80 nM T27812 CF3S2A 25109015 IC50 = 6900 nM T27812 CR86IN 25109441 IC50 = 720 nM T27812 C7N5TO 25118697 Ki = 17.7 nM T27812 CK58HA 25118698 Ki = 253 nM T27812 CFA5Y8 25118699 Ki = 22 nM T27812 CG2HJ3 25118700 Ki = 157 nM T27812 C08SZM 25119058 Ki = 8.3 nM T27812 C0OF5U 25119059 Ki = 262 nM T27812 C2MZB9 25119060 Ki = 2.4 nM T27812 CCE54T 25119061 Ki = 4.3 nM T27812 CM80TD 25119062 Ki = 8 nM T27812 C9RCX3 25119063 Ki = 3.8 nM T27812 CDEX47 25119406 Ki = 7.9 nM T27812 CXF1N0 25119407 Ki = 15.5 nM T27812 CL1GE2 25119409 Ki = 3.2 nM T27812 C0J3RD 25138742 IC50 = 379 nM T27812 C8SPL6 25138902 IC50 = 452 nM T27812 CSM12R 25138907 IC50 = 24.3 nM T27812 CN13MI 25138912 IC50 = 612 nM T27812 C3LHY5 25138913 IC50 > 1000 nM T27812 CGBL04 25139014 Ki = 1200 nM T27812 CTYC19 25139055 IC50 = 56.5 nM T27812 C9JR6E 25139058 IC50 = 28.3 nM T27812 C3VNW8 25139062 IC50 > 1000 nM T27812 C1QHJ5 25139063 IC50 = 776 nM T27812 CAY54E 25139064 IC50 > 1000 nM T27812 CB8E6J 25139065 IC50 = 138 nM T27812 C2L3OB 25139066 IC50 > 1000 nM T27812 C5PO7X 25139217 IC50 = 147 nM T27812 C0A5NK 25139366 IC50 = 47 nM T27812 C9RO2S 25139374 IC50 = 103 nM T27812 CS14YK 25139517 IC50 > 1000 nM T27812 C5JWI0 25139643 IC50 = 834 nM T27812 C6I9FN 25139645 IC50 > 1000 nM T27812 CJ63XC 25139652 IC50 > 1000 nM T27812 C6OCL8 25139785 IC50 = 435 nM T27812 CA3E2B 25139914 IC50 > 1000 nM T27812 CD69BU 25140055 IC50 > 1000 nM T27812 CP57TN 25140057 IC50 > 1000 nM T27812 CG05CH 25140362 IC50 = 193 nM T27812 CJ5VX0 25140466 Ki = 490 nM T27812 CQO5P0 25140648 IC50 = 15 nM T27812 C0YEI8 25141192 Ki = 535 nM T27812 C7W9YX 25150535 IC50 = 140 nM T27812 C35XQI 25150621 IC50 = 32 nM T27812 CD0QU5 25150624 IC50 = 45 nM T27812 CIZ1N9 25150625 IC50 = 16 nM T27812 C6IXV9 25150627 IC50 = 81 nM T27812 CE1ND3 25150628 IC50 = 26 nM T27812 CAVR45 25150711 IC50 = 97 nM T27812 CW9MX8 25168440 Ki = 2 nM T27812 CXC35U 25168857 IC50 = 800 nM T27812 C0YOQ7 25176461 IC50 = 6.8 nM T27812 C1JL9X 25176462 IC50 = 13 nM T27812 C30VBG 25181825 IC50 = 3100 nM T27812 C4W2AK 25181826 IC50 = 1100 nM T27812 C7JYI8 25188212 Ki = 430 nM T27812 C56CDP 25188770 Ki = 93 nM T27812 C5Z0LT 25188771 Ki = 463 nM T27812 C46ANM 25195291 Ki = 4440 nM T27812 C37YTG 25210603 Ki = 0.3981 nM T27812 CW3JR1 25210604 Ki = 1 nM T27812 CCTO39 25210872 Ki = 0.2512 nM T27812 CE7BA0 25210873 Ki = 0.631 nM T27812 C0FE8U 25210874 Ki = 0.5012 nM T27812 C0XN3L 25210876 Ki = 0.3162 nM T27812 CF6AD3 25211583 IC50 = 42 nM T27812 CVU7J1 25211682 Ki = 65 nM T27812 C2E6QB 25212170 Ki > 10000 nM T27812 CJ1Z9H 25216680 Ki = 300 nM T27812 C1T3LR 25218143 Ki = 170 nM T27812 CPI03N 25218397 Ki > 3000 nM T27812 CL1R3Q 25218401 Ki = 810 nM T27812 CX07CK 25258806 IC50 > 100000 nM T27812 CHY8S9 25258809 IC50 = 18.4 nM T27812 C3F0CJ 25260132 IC50 = 554 nM T27812 C7PK2X 29938807 Ki = 42 nM T27812 CSO5Y3 29981497 Ki = 63900 nM T27812 CN8J0W 29981513 Ki > 10000000 nM T27812 CJ1N0X 29981679 Ki = 266000 nM T27812 CH3M1E 31413243 IC50 > 10000 nM T27812 C9GS1N 31413320 IC50 > 10000 nM T27812 C2XY4V 31413484 IC50 > 10000 nM T27812 CW2KO7 31568498 IC50 = 230 nM T27812 CHE3I4 33139722 IC50 > 10000 nM T27812 C4FR6G 36465568 IC50 > 10000 nM T27812 CRD0C3 42273320 IC50 = 4460 nM T27812 C2TUQ3 42273630 IC50 = 280 nM T27812 C7C9DY 42629242 IC50 = 3 nM T27812 C1J4XZ 42636222 IC50 = 3380 nM T27812 CR70ZY 43164282 IC50 = 201 nM T27812 C0AI7N 43229249 Ki = 1534 nM T27812 CK0C3Z 43282996 IC50 = 13.9 nM T27812 C2VNA3 43283055 IC50 = 12.8 nM T27812 CNL52R 43283283 IC50 = 56 nM T27812 C6P5DK 43283415 IC50 = 18 nM T27812 CP16RL 43285101 IC50 = 94.1 nM T27812 C0VC7J 43314210 IC50 = 7.55 nM T27812 CYV94L 43314375 IC50 = 5.53 nM T27812 C1YM3D 44131466 Ki = 887 nM T27812 CMTB93 44131470 Ki = 30 nM T27812 CYE20L 44131666 Ki > 4710 nM T27812 CPR7L3 44133672 Ki = 203 nM T27812 CE3SD9 44133859 Ki = 2 nM T27812 CZ2VQ1 44133861 Ki = 2.7 nM T27812 C9P5XU 44133863 Ki = 36 nM T27812 C2G7AO 44134036 Ki = 102 nM T27812 C5YKI9 44134038 Ki = 194 nM T27812 C6DQJ3 44134039 Ki = 1850 nM T27812 C8RZX0 44134041 Ki = 109 nM T27812 CXZH39 44138098 Ki = 316.23 nM T27812 CUOD42 44138104 Ki = 10 nM T27812 CW5Q9P 44143473 Ki = 1.1 nM T27812 CO0GC4 44157259 Ki > 6000 nM T27812 CGA8B4 44157339 Ki > 6000 nM T27812 C25DHI 44178203 Ki = 1.995 nM T27812 C8R1QU 44178224 Ki = 0.67 nM T27812 CW3X1D 44182545 Ki = 3.37 nM T27812 CI8SO3 44182695 Ki = 1.17 nM T27812 CQP5G0 44182696 Ki = 5.25 nM T27812 CYMQ43 44182839 Ki = 5.32 nM T27812 CI12UH 44188274 IC50 = 109 nM T27812 CT30BL 44188275 IC50 = 7 nM T27812 CH7FJ6 44188689 Ki = 15.85 nM T27812 CSE8X3 44188690 Ki = 6.31 nM T27812 CY2Q9O 44188691 Ki = 31.62 nM T27812 C6FPM5 44188693 Ki = 3.981 nM T27812 CWR04I 44188695 Ki = 5.012 nM T27812 CJEG24 44188861 Ki = 19.95 nM T27812 C9XSI6 44189029 Ki = 15.85 nM T27812 C2AV1K 44190762 IC50 = 970 nM T27812 CY6KC3 44194561 Ki = 0.013 nM T27812 C6WSI1 44204599 IC50 = 108.4 nM T27812 C2KJB0 44216880 Ki = 0.4 nM T27812 CA50PK 44219207 Ki = 0.3981 nM T27812 CQY1J3 44219363 Ki = 1.995 nM T27812 CJX5T2 44219364 Ki = 0.7943 nM T27812 C6SF0L 44219365 Ki = 1 nM T27812 CWP84D 44219367 Ki = 0.7943 nM T27812 CVG5I0 44219517 Ki = 5.012 nM T27812 C1NQ2R 44219519 Ki = 0.631 nM T27812 CKMV39 44219520 Ki = 3.162 nM T27812 CA46YO 44230734 Ki = 34 nM T27812 CCK73R 44230855 IC50 = 530 nM T27812 CB5P7N 44230873 Ki = 53 nM T27812 CXI7Z8 44230875 Ki = 13 nM T27812 CU8MS7 44230877 Ki = 66 nM T27812 C67PRE 44231009 Ki = 8 nM T27812 C67WIP 44231010 Ki = 871 nM T27812 CCP13S 44231144 Ki = 1 nM T27812 CIBR82 44231149 Ki = 13 nM T27812 CE12BT 44231265 Ki = 22 nM T27812 C0TF4H 44231266 Ki = 4 nM T27812 C7HCZ5 44231267 Ki = 66 nM T27812 CDZ8F4 44231268 Ki = 41 nM T27812 C0AW6X 44241240 IC50 = 570 nM T27812 C8AFN4 44241291 IC50 = 200 nM T27812 C63GVH 44241292 IC50 = 88 nM T27812 CL09IQ 44263496 IC50 > 10000 nM T27812 C87MXH 44263497 IC50 > 10000 nM T27812 C8WZG7 44269522 Ki = 0.08 nM T27812 C0MCK3 44269548 Ki = 1.35 nM T27812 C96ZRI 44269549 Ki = 0.11 nM T27812 C5YE8A 44269598 Ki = 0.08 nM T27812 CI14GD 44269607 Ki = 0.04 nM T27812 CE20CZ 44275807 Ki = 3548.13 nM T27812 C1QHI4 44295709 IC50 = 2.53 nM T27812 C2B8AN 44295896 IC50 = 1 nM T27812 CC3T9P 44295975 Ki = 4 nM T27812 C5S1ZP 44297545 IC50 = 133 nM T27812 CTNB69 44297557 IC50 = 49.9 nM T27812 C40LQR 44297587 IC50 = 4970 nM T27812 CAX8D2 44297669 IC50 = 19.7 nM T27812 CS5H4Y 44297830 IC50 = 1073 nM T27812 CM58FQ 44297831 IC50 = 550 nM T27812 CV3PH7 44299504 Ki = 51.16 nM T27812 C0OX9M 44299511 Ki = 1.99 nM T27812 COI7M3 44299729 Ki = 12.63 nM T27812 CEO46F 44305466 Ki = 2330 nM T27812 C97SYT 44305491 Ki = 0.56 nM T27812 CZG6F3 44305492 Ki = 42 nM T27812 CD3M2K 44307360 Ki = 38.6 nM T27812 CUSR03 44307440 Ki = 1.23 nM T27812 C3WLT2 44307441 Ki = 74.1 nM T27812 C7U8NC 44307585 Ki = 55.1 nM T27812 C8RHD9 44308474 Ki = 102.3 nM T27812 C0LCV4 44308475 IC50 = 176 nM T27812 C0O2BH 44308682 Ki = 357 nM T27812 C0UDG4 44313303 Ki = 92 nM T27812 C1P0XE 44316740 Ki = 1.15 nM T27812 C62EYI 44316755 Ki = 13.59 nM T27812 CVKF37 44316789 Ki = 14.71 nM T27812 CFK6D0 44316790 Ki = 0.27 nM T27812 COM46U 44316963 Ki = 0.44 nM T27812 C2PB8C 44317057 Ki = 1.1 nM T27812 CXOP69 44317095 Ki = 0.58 nM T27812 CL78IT 44317121 Ki = 0.31 nM T27812 CBMS83 44317146 Ki = 0.51 nM T27812 C38IFX 44321638 IC50 > 10000 nM T27812 CX1EB8 44322005 IC50 = 180 nM T27812 C1B4LU 44322022 IC50 = 9560 nM T27812 CV7NH3 44322023 IC50 = 2520 nM T27812 C7S2VP 44322076 IC50 > 10000 nM T27812 CI0GO4 44322143 IC50 = 3320 nM T27812 CQHJ59 44322164 IC50 > 10000 nM T27812 CI90PQ 44322194 IC50 > 20000 nM T27812 CBN85G 44322218 IC50 = 28600 nM T27812 CGA75L 44322219 IC50 > 10000 nM T27812 CV1Q8O 44322257 IC50 = 5.57 nM T27812 CLY2O1 44322269 IC50 = 5820 nM T27812 CH0T6J 44322276 IC50 = 166 nM T27812 C9APJ1 44322284 IC50 = 677 nM T27812 CP21ST 44322286 IC50 = 4850 nM T27812 C5DVG7 44322287 IC50 = 991 nM T27812 CU7R1K 44322314 IC50 = 533 nM T27812 CB4V5Y 44322477 IC50 = 10700 nM T27812 CNMH73 44322592 IC50 = 15 nM T27812 CLE8Z7 44322610 Ki = 251.19 nM T27812 CG5L9Y 44322645 IC50 > 10000 nM T27812 C0PXM6 44322646 IC50 > 100000 nM T27812 C02LRC 44322770 Ki = 16.75 nM T27812 CW2P4D 44323130 Ki = 0.3 nM T27812 CQ4C8I 44323137 Ki = 1.69 nM T27812 CPB3U4 44323179 Ki = 4.35 nM T27812 CE1T8P 44323347 IC50 = 3530 nM T27812 CW16JD 44324737 Ki = 1.7 nM T27812 CA84SN 44324765 Ki = 1.2 nM T27812 COA3H4 44324800 Ki = 2.3 nM T27812 CY04JW 44324972 Ki = 4.5 nM T27812 CV7L8H 44330114 Ki = 22 nM T27812 C7Q1HP 44330168 Ki = 74 nM T27812 COY19U 44330368 Ki = 7.6 nM T27812 C1Z6DB 44330369 Ki = 4.8 nM T27812 CKO67I 44330427 Ki = 7.1 nM T27812 CP7Y9I 44330571 Ki = 35 nM T27812 C3AY4O 44330584 Ki = 13 nM T27812 CVTA63 44330598 Ki = 2.5 nM T27812 C83NZA 44330609 Ki = 5.6 nM T27812 C2AOH6 44330617 Ki = 0.6 nM T27812 C2RQ3Z 44330621 Ki = 1.3 nM T27812 C7JP2X 44330635 Ki = 1.6 nM T27812 CCVE83 44330645 Ki = 21 nM T27812 CO8XC7 44330653 Ki = 2.7 nM T27812 C47ZPQ 44330668 Ki = 1.9 nM T27812 CGJ05Y 44330679 Ki = 63 nM T27812 C9D2SN 44330857 Ki = 51 nM T27812 C5VN6Y 44332279 IC50 > 20000 nM T27812 CU0SQ8 44332340 IC50 = 251 nM T27812 C1E9NU 44332360 IC50 = 1310 nM T27812 C6F4XC 44332405 IC50 = 106 nM T27812 C78AWT 44332801 IC50 = 147 nM T27812 CEG5D6 44332819 IC50 = 68 nM T27812 C6BJZ0 44335519 Ki = 93.6 nM T27812 C5JCR2 44335674 Ki = 127.8 nM T27812 C7OW8Y 44336061 Ki = 532 nM T27812 CICR35 44340153 Ki = 12 nM T27812 CJL61A 44340169 Ki = 3.6 nM T27812 C40RKF 44340181 Ki = 2.3 nM T27812 C78CFJ 44340203 Ki = 5.8 nM T27812 CB34ZC 44340445 Ki = 25 nM T27812 CVWM21 44340483 Ki = 2.6 nM T27812 C4TSF5 44340484 Ki = 47 nM T27812 CQL94N 44340485 Ki = 4.4 nM T27812 C51NOI 44344091 Ki = 3118000 nM T27812 CX12US 44344115 Ki = 31700 nM T27812 C4PT6K 44344218 Ki = 3660 nM T27812 CX2O9B 44344235 Ki = 9600 nM T27812 C47SLT 44348860 IC50 = 3440 nM T27812 C1A2DC 44348878 IC50 = 9280 nM T27812 CQ54ET 44348881 IC50 = 21000 nM T27812 C5B8PU 44348886 IC50 = 4390 nM T27812 CZU4K0 44348893 IC50 = 10100 nM T27812 CQ7FV5 44348898 IC50 = 234 nM T27812 C1UQ8B 44348903 IC50 = 2430 nM T27812 C97XUW 44348914 IC50 = 550 nM T27812 CD5I2E 44348915 IC50 = 2200 nM T27812 C7PFJ2 44348927 IC50 = 19.7 nM T27812 CV8GJ6 44348934 IC50 = 9800 nM T27812 CFQ6K0 44348935 IC50 = 4930 nM T27812 C95ESH 44348942 IC50 = 4970 nM T27812 CX78DN 44348951 IC50 = 5960 nM T27812 CV9LR5 44348952 IC50 = 13200 nM T27812 CS3UM7 44349165 IC50 = 8550 nM T27812 CU9VM1 44349166 IC50 = 3360 nM T27812 C91DNF 44349181 IC50 = 5770 nM T27812 C03RQI 44351345 Ki = 0.24 nM T27812 C43ZES 44351406 Ki = 0.53 nM T27812 CO5G7D 44351470 Ki = 0.86 nM T27812 CCI5T8 44354020 Ki > 10000 nM T27812 CGQ13N 44354021 Ki = 168 nM T27812 C68QVH 44354105 Ki = 271 nM T27812 C2TGL8 44354122 Ki > 10000 nM T27812 C4GVC5 44354236 IC50 = 23 nM T27812 CFW7N2 44358674 IC50 = 71.8 nM T27812 CUN25S 44358675 IC50 = 28.5 nM T27812 C7BRY8 44358948 Ki = 2.4 nM T27812 CC6E7V 44358977 Ki = 2.3 nM T27812 CYI70C 44358978 Ki = 4 nM T27812 CYL37V 44358996 Ki = 2.1 nM T27812 CNU16S 44358997 Ki = 2 nM T27812 CWP87F 44359029 Ki = 19 nM T27812 C0HTE7 44359122 Ki = 7.6 nM T27812 C51KZA 44359123 Ki = 14.5 nM T27812 CL03NH 44359135 Ki = 10 nM T27812 CA1Q4M 44359155 Ki = 3.5 nM T27812 CS6O4C 44359156 Ki = 2.2 nM T27812 CDCU47 44359185 Ki = 3.8 nM T27812 CI0OX3 44359318 Ki = 4.1 nM T27812 CC2W7X 44359319 Ki = 0.95 nM T27812 C48UAD 44359478 Ki = 31 nM T27812 CJ36NW 44364204 Ki = 130 nM T27812 C0O2NU 44364206 Ki = 2.4 nM T27812 CMA5D4 44364314 Ki = 380 nM T27812 C69BCI 44364358 Ki = 500 nM T27812 CL2M6Y 44364359 Ki = 4.7 nM T27812 C35MGZ 44364439 Ki = 2100 nM T27812 CLW8D9 44364455 Ki = 2 nM T27812 CH26LQ 44365682 Ki = 8.5 nM T27812 C1M0OB 44365720 Ki = 33 nM T27812 C7QAW8 44365737 Ki = 4.69 nM T27812 C10HST 44365811 Ki = 26 nM T27812 CRY94A 44370219 IC50 = 1240 nM T27812 CTB3Q6 44372823 Ki = 0.67 nM T27812 C5DA8L 44372825 Ki = 427 nM T27812 CWGQ58 44383909 Ki = 0.05 nM T27812 CP4JB9 44384015 IC50 = 1.3 nM T27812 CU8Z1R 44384016 IC50 = 1.15 nM T27812 C24DSJ 44384117 Ki = 1.15 nM T27812 CC0XH9 44384512 IC50 = 0.32 nM T27812 CI52GK 44387798 Ki = 61 nM T27812 CQT45N 44390371 IC50 = 1100 nM T27812 C13WMU 44390389 IC50 = 2 nM T27812 C8YGL6 44390396 Ki = 4 nM T27812 C8IB4F 44390397 IC50 = 7 nM T27812 C51PVM 44390408 IC50 = 31 nM T27812 C31JQX 44390410 IC50 = 29 nM T27812 CFM14N 44390419 IC50 = 36 nM T27812 C0VB9N 44390420 IC50 = 32 nM T27812 C7DT6S 44391257 Ki = 50.12 nM T27812 C0UEV5 44391270 Ki = 79.43 nM T27812 CD2ZS6 44391745 IC50 = 11 nM T27812 C0NJZ3 44393374 IC50 = 180 nM T27812 CUI1Y3 44393424 IC50 = 77 nM T27812 C79ZVN 44393433 IC50 = 110 nM T27812 C71TRU 44393437 IC50 = 150 nM T27812 C73YHL 44393445 IC50 = 82 nM T27812 C7PYQ8 44393454 IC50 = 250 nM T27812 CAYF72 44393458 IC50 = 510 nM T27812 CUJV45 44393464 IC50 = 59 nM T27812 CFOL40 44393469 IC50 = 410 nM T27812 CZT98U 44393470 IC50 = 5.5 nM T27812 C8XLI0 44393483 IC50 = 54 nM T27812 C93ONE 44393487 IC50 = 430 nM T27812 C8CP6S 44393494 IC50 = 73 nM T27812 C64HWN 44393498 IC50 = 92 nM T27812 CGP92T 44393507 IC50 = 100 nM T27812 CJL5G2 44393519 IC50 = 400 nM T27812 C1YK0X 44393525 IC50 = 45 nM T27812 CD57ME 44393526 IC50 = 91 nM T27812 CHT8C4 44393532 IC50 = 140 nM T27812 C0X1EF 44393533 IC50 = 23 nM T27812 CGT4W1 44393595 IC50 = 480 nM T27812 CD9A7M 44393597 IC50 = 5 nM T27812 C1BXI7 44395690 IC50 = 700 nM T27812 CEY74D 44395805 IC50 = 28000 nM T27812 CZWE51 44395806 IC50 > 10000 nM T27812 C7ZGQ3 44395831 IC50 > 10000 nM T27812 CY2WM9 44395924 IC50 = 1300 nM T27812 CX0V4W 44398372 Ki = 0.57 nM T27812 CA09EW 44404169 Ki > 100 nM T27812 C5Y8LB 44404175 Ki > 100 nM T27812 CM46ID 44404176 Ki > 100 nM T27812 CX02GP 44404182 Ki > 100 nM T27812 CV39CT 44404223 Ki = 160 nM T27812 CG4P9S 44404235 Ki > 100 nM T27812 C4E6QN 44404238 Ki > 100 nM T27812 CVW0P1 44404239 Ki = 128 nM T27812 CZ9GU0 44404250 Ki > 100 nM T27812 CF8Z6A 44404254 Ki > 100 nM T27812 CN15FZ 44404255 Ki > 100 nM T27812 C30QXS 44404259 Ki > 100 nM T27812 C8U9NH 44404261 Ki > 100 nM T27812 CRSC86 44404262 Ki > 100 nM T27812 CM7W1J 44404265 Ki > 100 nM T27812 CFP8D2 44404266 Ki > 100 nM T27812 C97CAH 44404269 Ki > 100 nM T27812 C5R7XB 44404273 Ki > 100 nM T27812 C5F2VA 44404274 Ki > 100 nM T27812 CGN87C 44404278 Ki > 100 nM T27812 CSO98W 44404279 Ki > 100 nM T27812 CRIG21 44404285 Ki > 100 nM T27812 CO57NJ 44404286 Ki > 100 nM T27812 C4Q2BS 44404551 IC50 = 120 nM T27812 CL6C2S 44404914 IC50 = 270 nM T27812 CSDN32 44405146 Ki = 705 nM T27812 C4DFS7 44405156 Ki = 227 nM T27812 CZI0A4 44405840 IC50 = 0.003 nM T27812 CR30FO 44405845 IC50 = 690 nM T27812 C9TUH6 44405846 IC50 = 1710 nM T27812 CFT43Y 44405871 IC50 = 16100 nM T27812 CS2Q0A 44405875 IC50 = 670 nM T27812 CR06US 44405876 IC50 = 72.6 nM T27812 CG3WT6 44405893 IC50 = 2570 nM T27812 CDF9N4 44405897 IC50 = 2520 nM T27812 C4GN3T 44405898 IC50 = 3770 nM T27812 CA3I0W 44407714 Ki > 10000 nM T27812 CIH46L 44408412 Ki = 4.15 nM T27812 CK6O7A 44408415 IC50 > 100 nM T27812 CV3QD5 44408434 Ki = 10.28 nM T27812 C7T6WF 44408435 IC50 > 100 nM T27812 CJ3NS2 44408441 IC50 > 100 nM T27812 CT52PU 44408442 IC50 > 100 nM T27812 CDQ34O 44408477 IC50 > 100 nM T27812 CI3Z8X 44408529 IC50 > 100 nM T27812 CYP8A5 44408580 IC50 > 100 nM T27812 CA3P6K 44408581 IC50 > 100 nM T27812 C6F5EC 44408582 IC50 > 100 nM T27812 CKX2P8 44408664 IC50 = 5 nM T27812 C3C9PW 44408718 IC50 = 3 nM T27812 CK9U7V 44408719 IC50 = 2 nM T27812 C83DCF 44408748 IC50 = 6 nM T27812 CQ64UC 44408749 IC50 = 7 nM T27812 C14BYG 44408753 IC50 = 10 nM T27812 CI0JZ2 44408756 IC50 = 3 nM T27812 C9U3TR 44408757 IC50 = 10 nM T27812 C6LTD5 44408760 IC50 = 4 nM T27812 CYAC79 44408761 IC50 = 6 nM T27812 CX2S0E 44408762 IC50 = 1 nM T27812 C3QCP2 44408802 IC50 = 54 nM T27812 CLJ3U7 44408856 IC50 = 13 nM T27812 C5K8NB 44408857 IC50 = 25 nM T27812 C2QMD8 44408858 IC50 = 7 nM T27812 CI3ZS8 44408859 IC50 = 60 nM T27812 C1ZPY7 44408870 IC50 = 8 nM T27812 C8ZH4C 44408871 IC50 = 31 nM T27812 CB7WI1 44408872 IC50 = 140 nM T27812 C2J1KW 44408875 IC50 = 2 nM T27812 CZ8G2B 44408876 IC50 = 6 nM T27812 CR8KL1 44408880 IC50 > 1000 nM T27812 CKR78J 44408885 IC50 = 24 nM T27812 CC9D8S 44408886 IC50 = 65 nM T27812 CW7VA3 44408917 IC50 = 5 nM T27812 CBS73M 44408918 IC50 = 31 nM T27812 CE06JR 44408920 IC50 = 90 nM T27812 CQ45GH 44408921 IC50 = 30 nM T27812 CKM7O2 44408922 IC50 = 340 nM T27812 C13IEG 44408925 IC50 = 290 nM T27812 CE5AC6 44408926 IC50 = 240 nM T27812 C2D5WU 44408969 IC50 = 25 nM T27812 CG87PW 44409290 Ki > 1000 nM T27812 C24AHO 44411099 Ki = 0.48 nM T27812 C2EQ1I 44411140 Ki = 1.5 nM T27812 CCBK16 44411148 Ki = 2.2 nM T27812 C7D8MV 44411168 Ki = 6.8 nM T27812 CDH1U9 44411170 Ki = 3.6 nM T27812 C5Z3ES 44411177 Ki = 6.9 nM T27812 C60ECT 44411185 Ki = 1.9 nM T27812 CY0U6V 44411206 Ki = 0.28 nM T27812 CI6B1W 44411208 Ki = 0.39 nM T27812 C9GW7B 44411217 Ki = 4.1 nM T27812 C1R3LU 44411219 Ki = 1.4 nM T27812 C3M7RB 44411224 Ki = 0.96 nM T27812 C0J6WV 44411226 Ki = 0.48 nM T27812 CT7D0B 44411228 Ki = 0.3 nM T27812 C7TH4P 44411230 Ki = 1.1 nM T27812 C5FYQ9 44411235 Ki = 2.1 nM T27812 CI8MC6 44411239 Ki = 2.8 nM T27812 CFUV50 44411241 Ki = 3 nM T27812 CUFD63 44411249 Ki = 0.4 nM T27812 C9BV1K 44411254 Ki = 4.2 nM T27812 CM6RO7 44411258 Ki = 2.5 nM T27812 CE5A4F 44411296 Ki = 4.3 nM T27812 CR3P8E 44411314 Ki = 2.8 nM T27812 C8GD7M 44411395 Ki = 1.6 nM T27812 C42XFV 44411397 Ki = 1.1 nM T27812 CHU4D8 44411449 Ki = 0.26 nM T27812 CTO82V 44411451 Ki = 0.07 nM T27812 CWN14V 44411456 Ki = 1.5 nM T27812 CIG3V6 44411460 Ki = 2.5 nM T27812 CW3KE8 44411466 Ki = 1.5 nM T27812 CTQ19K 44411482 Ki = 1.2 nM T27812 C5ZN4X 44411491 Ki = 3.1 nM T27812 CV2S7W 44411499 Ki = 9.6 nM T27812 C6CW9U 44411501 Ki = 5.8 nM T27812 CC5Z7V 44411505 Ki = 2.2 nM T27812 C6OS1M 44411507 Ki = 15 nM T27812 CH8W2F 44411510 Ki = 0.8 nM T27812 CF4O1I 44411514 Ki = 7.9 nM T27812 C21MSX 44411516 Ki = 2.2 nM T27812 C4DZ1I 44411518 Ki = 8 nM T27812 CW0DM3 44411520 Ki = 2.2 nM T27812 C9JXM6 44411522 Ki = 0.7 nM T27812 C0DHC7 44411524 Ki = 3.1 nM T27812 CU8M4K 44411526 Ki = 1.3 nM T27812 C8XF4A 44411527 Ki = 0.8 nM T27812 C6PR1D 44411536 Ki = 4 nM T27812 C2GV3H 44411541 Ki = 17 nM T27812 CDI7R3 44411543 Ki = 5 nM T27812 CIBG87 44413825 Ki > 2000 nM T27812 CFN48L 44413826 Ki = 1.9 nM T27812 CA97VC 44413836 Ki = 290 nM T27812 CLG5H8 44413837 Ki > 2000 nM T27812 CCY43Q 44413856 Ki = 1230 nM T27812 CW0VE9 44413857 Ki = 1650 nM T27812 C05UKL 44413866 IC50 > 2000 nM T27812 CCJ4X1 44413903 Ki > 2000 nM T27812 C81IAE 44413904 Ki = 94 nM T27812 C5Z2GC 44413925 Ki = 110 nM T27812 C3BMI9 44413953 IC50 > 2000 nM T27812 C18JHP 44413959 Ki = 513 nM T27812 C3IE4V 44414667 IC50 > 400 nM T27812 CQ3C7F 44414684 IC50 > 400 nM T27812 CNR87Z 44414690 IC50 = 15 nM T27812 CCL7Y9 44414691 IC50 = 28 nM T27812 CM9V8F 44414692 IC50 = 13 nM T27812 CQD2S5 44414696 IC50 = 13 nM T27812 CM6D5P 44414704 IC50 = 17 nM T27812 CZ9LM3 44414707 IC50 = 10 nM T27812 CE85AH 44414731 IC50 = 39 nM T27812 C2BYE0 44414733 IC50 = 13 nM T27812 C9XIR1 44414734 IC50 = 38 nM T27812 C9FCZ2 44414748 IC50 = 12 nM T27812 C8RN6K 44414749 IC50 = 40 nM T27812 C81QHB 44414760 IC50 = 11 nM T27812 CV37KC 44414761 IC50 = 8.2 nM T27812 CUK97V 44414762 IC50 = 30 nM T27812 CI8NH6 44414763 IC50 = 10 nM T27812 C3LJ7N 44414780 IC50 = 12 nM T27812 CY5Q9A 44414800 IC50 = 14 nM T27812 C3RZ0N 44414809 IC50 = 46 nM T27812 CPR9Y5 44414810 IC50 = 79 nM T27812 CF8Q6Y 44414836 IC50 = 9.8 nM T27812 CWZ3E4 44414859 IC50 = 42 nM T27812 CA58NQ 44414873 IC50 = 300 nM T27812 CHCQ59 44414875 IC50 = 3.9 nM T27812 CVTQ68 44416033 Ki = 0.28 nM T27812 CZ6WJ8 44416034 Ki = 0.82 nM T27812 CRA8M1 44416084 Ki = 0.09 nM T27812 C1BF0K 44416103 Ki = 98.31 nM T27812 C9Q5UZ 44416104 Ki = 5.63 nM T27812 C9UDS3 44416105 Ki = 18.75 nM T27812 CHF6L7 44417598 Ki = 0.2 nM T27812 CK5PZ8 44417599 Ki = 0.2 nM T27812 CRZK78 44418862 IC50 = 1100 nM T27812 CXA51W 44419295 Ki = 40 nM T27812 CLA67J 44419296 Ki = 212 nM T27812 C82VQX 44419298 Ki = 11 nM T27812 CRAK93 44419299 Ki = 710 nM T27812 CZT81O 44419300 Ki = 49 nM T27812 C2WDJ5 44419301 Ki = 305 nM T27812 C85OTF 44419303 Ki = 328 nM T27812 CZ5O8Y 44419306 Ki = 5465 nM T27812 CXP1A6 44419308 Ki = 224 nM T27812 CM3K1F 44419314 Ki = 35 nM T27812 CG8F3J 44419327 Ki = 42 nM T27812 CJR7P1 44419328 Ki = 18 nM T27812 C7DQL6 44419331 Ki = 3.5 nM T27812 CVMF25 44419335 Ki = 117 nM T27812 C59ZPV 44419340 Ki = 217 nM T27812 C71CPW 44419344 Ki = 166 nM T27812 CM1WZ9 44419345 Ki = 69 nM T27812 CJHN07 44421413 Ki = 518 nM T27812 CEHO31 44421414 Ki = 460 nM T27812 C2WE3K 44421423 Ki = 20.6 nM T27812 C1S3RH 44421438 Ki = 441 nM T27812 CSIN57 44421439 IC50 > 2000 nM T27812 CQI4V3 44421455 Ki = 390 nM T27812 C2BEZ9 44421482 Ki = 910 nM T27812 C7PCA5 44421483 Ki = 410 nM T27812 CNYK42 44421484 Ki = 1250 nM T27812 CB17LT 44421485 Ki = 1470 nM T27812 CE6G3H 44421486 Ki = 25 nM T27812 CL6M9V 44421497 Ki = 100 nM T27812 CSU23Q 44421500 Ki = 4100 nM T27812 CL1V7W 44422784 IC50 = 3 nM T27812 CK7HF3 44424855 Ki = 2.1 nM T27812 CV43NH 44427225 IC50 = 2000 nM T27812 CGX49R 44427889 Ki = 0.08 nM T27812 C7I2MZ 44427901 Ki = 0.08 nM T27812 CGOD89 44429174 Ki = 1850 nM T27812 C6BW5V 44429184 Ki = 2810 nM T27812 CIJ5R2 44429185 Ki = 217 nM T27812 C6OVA2 44429187 Ki = 3000 nM T27812 CNP37Y 44429189 Ki = 785000 nM T27812 C8SR0G 44429190 Ki = 2840000 nM T27812 C53AFL 44429191 Ki = 2240000 nM T27812 CN4UT8 44429192 Ki = 417000 nM T27812 C5HK8Y 44429193 Ki = 2690000 nM T27812 C7J6GA 44429194 Ki = 1460000 nM T27812 CK9H1C 44429195 Ki = 3800000 nM T27812 CPB4D3 44429196 Ki = 3388000 nM T27812 CQA0W7 44429197 Ki = 296000 nM T27812 CV9M4N 44429198 Ki = 1950000 nM T27812 CUH0B6 44429199 Ki = 1141000 nM T27812 CS2ER7 44429200 Ki = 228000 nM T27812 CE2M3T 44429201 Ki = 1860000 nM T27812 CE31CZ 44429202 Ki = 1180000 nM T27812 CF5CO6 44429203 Ki = 109000 nM T27812 CJ9VZ1 44429204 Ki = 841000 nM T27812 CJ5F4X 44429205 Ki = 2250000 nM T27812 CLK84J 44429206 Ki = 4680000 nM T27812 CH50DU 44429207 Ki = 668000 nM T27812 C1Z7KB 44429209 Ki = 5020000 nM T27812 C7OQT6 44429210 Ki = 4710000 nM T27812 CI46CX 44429212 Ki = 573000 nM T27812 CA2HN0 44429214 Ki = 28700 nM T27812 CE30YG 44429218 Ki = 149000 nM T27812 CM5HG8 44429219 Ki = 706000 nM T27812 C4I1GO 44429221 Ki = 463000 nM T27812 CDGP34 44429222 Ki = 532000 nM T27812 CW7L3V 44429226 Ki = 32000 nM T27812 CKF60U 44429227 Ki = 381000 nM T27812 CX4EM1 44429392 Ki = 390000 nM T27812 C3JNX9 44429393 Ki = 9120000 nM T27812 CH9W4Z 44429395 Ki = 605000 nM T27812 C3O9DN 44429396 Ki = 1510000 nM T27812 CO29HT 44429397 Ki = 1910000 nM T27812 C75HYO 44429399 Ki = 185000 nM T27812 C7TXV4 44429400 Ki = 73000 nM T27812 CBR73H 44429401 Ki = 1800000 nM T27812 CG9N0T 44429402 Ki = 1040000 nM T27812 C2JOU8 44430356 Ki = 2.9 nM T27812 C90VJB 44430358 Ki = 7.3 nM T27812 CBOP25 44430359 Ki = 3.4 nM T27812 CD0E3S 44430363 Ki = 19.3 nM T27812 C01VKH 44430365 Ki = 9.7 nM T27812 C4T7KP 44430367 Ki = 2 nM T27812 CZB0W3 44430368 Ki = 1.8 nM T27812 C1Z6WS 44430371 Ki = 18 nM T27812 C4KA7J 44430373 Ki = 7.2 nM T27812 CDP69G 44430375 Ki = 8 nM T27812 CR1IT7 44430379 Ki = 5.3 nM T27812 CU1F0L 44430380 Ki = 4 nM T27812 C07PLN 44430381 Ki = 33 nM T27812 CQG41A 44430844 IC50 = 830 nM T27812 CF4BK0 44430849 IC50 = 0.56 nM T27812 C82VMO 44430851 IC50 = 0.4 nM T27812 CQJ6S7 44430852 IC50 = 1 nM T27812 CL01CO 44430853 IC50 = 14 nM T27812 CO80EL 44430855 IC50 = 5.3 nM T27812 CJ1UO5 44430856 IC50 = 19 nM T27812 CI9KT8 44430860 IC50 = 150 nM T27812 CH2F3S 44430861 IC50 = 770 nM T27812 CL59HA 44431531 Ki = 0.8 nM T27812 C6JK5A 44431532 Ki = 3 nM T27812 C5LNH6 44431533 Ki = 7.4 nM T27812 CLX73C 44431534 Ki = 2.1 nM T27812 CCV62B 44431535 Ki = 8.1 nM T27812 C4P5XG 44431536 Ki = 2.2 nM T27812 CYPR70 44431537 Ki = 5.7 nM T27812 C6CD3M 44431728 Ki = 42.8 nM T27812 CT2UJ0 44431732 Ki = 136.29 nM T27812 CE2QP4 44431734 Ki = 4.16 nM T27812 CHR6F7 44431736 Ki = 9.04 nM T27812 CH6B3Y 44431739 Ki = 3.45 nM T27812 CZJ2W5 44434147 Ki = 2.5 nM T27812 CN8A3O 44434150 Ki = 6.7 nM T27812 CF42IC 44434165 Ki = 1.1 nM T27812 CY79ZO 44434236 Ki = 2.7 nM T27812 CCS8D1 44434250 Ki = 1.9 nM T27812 C4IF8K 44435317 Ki = 10.4 nM T27812 C0PRV8 44435318 Ki = 6.5 nM T27812 CGE72U 44437018 Ki > 50000 nM T27812 CFN21O 44437023 Ki > 50000 nM T27812 CVJ05I 44438666 Ki = 147 nM T27812 CF9R8D 44439854 Ki = 4.7 nM T27812 CS1LB8 44439855 Ki = 18 nM T27812 CDX7C5 44439856 Ki = 46 nM T27812 CY5J2W 44439857 Ki = 8.6 nM T27812 C10ZYB 44439858 Ki = 15 nM T27812 C3IJ7Y 44439859 Ki = 16 nM T27812 CHKE50 44439860 Ki = 13 nM T27812 CR1FY4 44439861 Ki = 34 nM T27812 CP9B4A 44439862 Ki = 13 nM T27812 C50ZDW 44439863 Ki = 13 nM T27812 CZ9F1A 44440497 Ki = 8 nM T27812 CZK1U5 44441058 Ki = 12.3 nM T27812 CF8K5H 44441067 Ki = 8.3 nM T27812 C6VC8I 44441070 Ki = 12.3 nM T27812 CFCO97 44441071 Ki = 18.7 nM T27812 C1O9VZ 44441073 Ki = 31.3 nM T27812 CI43TX 44441077 Ki = 2.7 nM T27812 CZOU36 44441079 Ki = 6 nM T27812 CV0UI9 44441083 Ki = 5 nM T27812 CITP46 44441084 Ki = 19.7 nM T27812 CX7N0I 44441085 Ki = 291 nM T27812 C69RCY 44441088 Ki = 121 nM T27812 CC0A8B 44441089 Ki = 119 nM T27812 C6P8RJ 44441332 IC50 = 4 nM T27812 CDEY23 44441334 IC50 = 6 nM T27812 COBN96 44441335 IC50 = 3 nM T27812 C23BGW 44441336 IC50 = 5 nM T27812 C92ABN 44441338 IC50 = 15 nM T27812 C6K8ZB 44441339 IC50 = 8 nM T27812 CJ2S0W 44441340 IC50 = 43 nM T27812 C1R0DN 44441341 IC50 = 9 nM T27812 C9FB6Y 44441345 IC50 = 5 nM T27812 CZ34LI 44441346 IC50 = 11 nM T27812 C2GAV7 44441348 IC50 = 13 nM T27812 CWH92R 44441349 IC50 = 11 nM T27812 C61VKY 44441350 IC50 = 24 nM T27812 CF4A8D 44441351 IC50 = 29 nM T27812 CD30KT 44441353 IC50 = 15 nM T27812 C8ZJU5 44443873 Ki > 500000 nM T27812 C4X5GY 44443875 Ki = 520000 nM T27812 CI0Q6D 44443877 Ki = 300000 nM T27812 COC4G7 44443878 Ki > 1000000 nM T27812 C9JB8C 44443887 Ki > 500000 nM T27812 C3Q8RJ 44443888 Ki = 540000 nM T27812 CCP50E 44443889 Ki > 500000 nM T27812 CSF8J3 44443890 Ki = 110000 nM T27812 CRB6J3 44443891 Ki = 24000 nM T27812 C0EI1N 44443892 Ki > 1000000 nM T27812 CZUT06 44443893 Ki = 500000 nM T27812 CWB8E6 44443894 Ki = 50000 nM T27812 CDW62E 44443895 Ki = 390000 nM T27812 CR1AP8 44443896 Ki > 1000000 nM T27812 CVK42D 44443897 Ki > 500000 nM T27812 CEI6Y9 44443898 Ki > 500000 nM T27812 C2WC8G 44443899 Ki = 910000 nM T27812 C03MYS 44443900 Ki = 24000 nM T27812 C53UET 44443988 IC50 = 25 nM T27812 CNA5S7 44444478 IC50 = 99 nM T27812 CZ47HL 44444488 IC50 = 410 nM T27812 C1VS2R 44444492 IC50 > 1000 nM T27812 C0YK4P 44444506 IC50 = 130 nM T27812 CXY41Z 44444512 IC50 > 1000 nM T27812 C3IMT5 44444513 IC50 = 89 nM T27812 C6FY0T 44444517 IC50 = 15 nM T27812 CHN6M7 44444520 IC50 = 58 nM T27812 CM53HC 44444521 IC50 = 120 nM T27812 C7I4XK 44444523 IC50 = 17 nM T27812 C09OBL 44444524 IC50 = 37 nM T27812 CMEO07 44444525 IC50 = 4.1 nM T27812 CDA23T 44444527 IC50 = 67 nM T27812 C1Z2VD 44444528 IC50 = 51 nM T27812 CVL6G4 44444529 IC50 = 16 nM T27812 C92VUT 44444530 IC50 = 48 nM T27812 CDAM09 44444532 IC50 = 52 nM T27812 CG0TP9 44444534 IC50 = 8.6 nM T27812 C46GMK 44444536 IC50 = 310 nM T27812 CO76LQ 44444537 IC50 = 550 nM T27812 CCMZ42 44444540 IC50 = 13 nM T27812 C5OSV3 44444542 IC50 = 5.9 nM T27812 C0YOW4 44448355 IC50 = 340 nM T27812 CZS5L9 44448356 IC50 = 1800 nM T27812 CG4D7J 44448357 IC50 = 320 nM T27812 C9RJX0 44448358 IC50 = 76 nM T27812 C7AW4C 44448387 IC50 = 84 nM T27812 C15HXQ 44448388 IC50 = 60 nM T27812 C1OQ2Y 44448389 IC50 = 40 nM T27812 CE80KR 44448391 IC50 = 47 nM T27812 CQV39U 44448392 IC50 = 34 nM T27812 CPV4Z3 44448423 IC50 = 590 nM T27812 CFC8I2 44448425 IC50 = 71 nM T27812 CM8QA0 44448426 IC50 = 47 nM T27812 C1LIQ2 44448427 IC50 = 76 nM T27812 CW51IM 44448465 IC50 = 140 nM T27812 C1MIQ3 44448466 IC50 = 60 nM T27812 CO4GZ7 44448467 IC50 > 10000 nM T27812 COE35W 44448468 IC50 = 3100 nM T27812 C5GTQ1 44448470 IC50 = 4400 nM T27812 CJ8X7A 44448508 IC50 = 9600 nM T27812 CKO0F9 44448509 IC50 = 290 nM T27812 C36MOD 44448511 IC50 = 4000 nM T27812 CCR7Q2 44448512 IC50 = 620 nM T27812 CPS91V 44448544 IC50 = 2200 nM T27812 CO9U4F 44448545 IC50 = 2000 nM T27812 CM6W2E 44448546 IC50 = 3500 nM T27812 CWA0E4 44448547 IC50 = 350 nM T27812 C9HVB8 44448548 IC50 = 520 nM T27812 CSYB74 44448582 IC50 = 520 nM T27812 CF0ZG2 44448584 IC50 = 65 nM T27812 C67GMI 44449234 IC50 = 10 nM T27812 C3RMF8 44449236 IC50 = 6 nM T27812 CM4F7Z 44449237 IC50 = 23 nM T27812 C2UQI1 44449238 IC50 = 4 nM T27812 C3HS9U 44449239 IC50 = 6 nM T27812 CQN4Z9 44449267 IC50 = 3 nM T27812 CZ3UA5 44449268 Ki = 13 nM T27812 C8FBZ0 44449269 IC50 = 14 nM T27812 CS6R9X 44449270 Ki = 18 nM T27812 CKH31F 44449272 IC50 = 11 nM T27812 CD4J9E 44449296 IC50 = 46 nM T27812 CGK7O1 44449297 IC50 = 6 nM T27812 CVZ39S 44449298 IC50 = 4 nM T27812 C2O9KI 44449307 IC50 = 270 nM T27812 C9MU1V 44449332 IC50 = 14 nM T27812 CJC38Z 44449333 IC50 = 7 nM T27812 C6X4JZ 44449340 IC50 = 430 nM T27812 CCB54W 44449341 IC50 = 1700 nM T27812 C1CPD4 44449368 IC50 = 32 nM T27812 CR4OB8 44449369 IC50 = 280 nM T27812 C7W4XU 44449370 IC50 = 2100 nM T27812 CC2ZK5 44449371 IC50 = 54 nM T27812 CZSE46 44449372 IC50 = 370 nM T27812 CZY4G7 44449373 IC50 = 1100 nM T27812 CH48QG 44449395 IC50 = 100 nM T27812 C2YG0E 44449396 IC50 = 39 nM T27812 CD9LA2 44449397 IC50 = 160 nM T27812 CWG79A 44449398 IC50 = 210 nM T27812 CW98KH 44449399 IC50 = 3400 nM T27812 CYM7I3 44449400 IC50 = 560 nM T27812 CK9UP5 44449401 IC50 = 6400 nM T27812 C8EJ1M 44449434 IC50 = 125 nM T27812 C6KR7N 44449435 IC50 > 10000 nM T27812 C59NSQ 44449436 IC50 > 10000 nM T27812 C2QF0K 44449437 IC50 > 10000 nM T27812 C2Z6IM 44449438 IC50 = 6900 nM T27812 CJL4G7 44449462 IC50 = 540 nM T27812 C50SKP 44449464 IC50 = 280 nM T27812 CT76PB 44449465 IC50 = 13 nM T27812 COU68C 44449519 IC50 = 112 nM T27812 C0X2RW 44449521 IC50 = 65 nM T27812 CG2AD9 44449552 IC50 = 140 nM T27812 CY0B5K 44449554 IC50 = 77 nM T27812 CHA59Q 44449589 IC50 = 28 nM T27812 CDQ89E 44449590 IC50 = 64 nM T27812 C53EYA 44449619 IC50 = 58 nM T27812 CUXK25 44449620 IC50 = 49 nM T27812 C7KZ5C 44449623 IC50 = 480 nM T27812 CZ1L4G 44449624 IC50 = 480 nM T27812 C8K3XF 44449625 IC50 = 150 nM T27812 CYRM03 44449651 IC50 = 210 nM T27812 C15DIZ 44449652 IC50 = 460 nM T27812 CWO0H5 44449656 IC50 = 145 nM T27812 C7ENK5 44449717 IC50 = 39 nM T27812 C41WXJ 44449718 IC50 = 8 nM T27812 C7KQ4B 44449719 IC50 = 24 nM T27812 CC5K0E 44449720 IC50 = 18 nM T27812 C2KA8J 44449721 IC50 = 231 nM T27812 C2QP0Z 44449729 IC50 = 130 nM T27812 C3VE2D 44449768 Ki = 22 nM T27812 C3FP2I 44449792 Ki = 740 nM T27812 C83ICG 44449794 Ki = 11 nM T27812 CS9ZO8 44449911 Ki = 60 nM T27812 C50ZLO 44449944 Ki = 240 nM T27812 CJ83BL 44450087 Ki = 69 nM T27812 CW9P8L 44450088 Ki = 88 nM T27812 CB8W3Q 44450089 Ki = 62 nM T27812 C26WAJ 44450090 Ki = 70 nM T27812 CMKF97 44450118 Ki = 70 nM T27812 C35FRM 44450119 Ki = 58 nM T27812 CK1B8X 44450120 Ki = 41 nM T27812 C4AUT7 44450121 Ki = 96 nM T27812 CJOI42 44450152 Ki = 110 nM T27812 C6FBZ1 44450153 Ki = 30 nM T27812 C52HPA 44450154 Ki = 20 nM T27812 C9SB0X 44450155 Ki = 100 nM T27812 CAW6S7 44450181 Ki = 12 nM T27812 CJ8KS4 44450182 Ki = 1800 nM T27812 C4M0PG 44450184 Ki = 34 nM T27812 C4KE7B 44450185 Ki = 3390 nM T27812 C4VL3W 44450211 Ki = 260 nM T27812 CSQR06 44450212 Ki = 20 nM T27812 CXR4G1 44450213 Ki = 185 nM T27812 CTX1Q7 44452747 Ki = 1420 nM T27812 CIS3J5 44452748 Ki = 218 nM T27812 COAL13 44452772 Ki = 265 nM T27812 C42KFD 44452774 Ki = 440 nM T27812 CGR0B6 44452775 Ki = 279 nM T27812 C80CWR 44452935 Ki = 4060 nM T27812 CY01KA 44452990 Ki = 2820 nM T27812 C8Q7OP 44452992 Ki = 821 nM T27812 CV92RP 44452994 Ki = 1470 nM T27812 CLSI34 44453016 Ki = 242 nM T27812 CKZN93 44453017 Ki = 1980 nM T27812 CB1OY5 44453042 Ki = 88 nM T27812 C2HFJ7 44453043 Ki = 384 nM T27812 CY38AM 44453067 Ki = 133 nM T27812 CBP25X 44453068 Ki = 235 nM T27812 CR4F7O 44453093 Ki = 136 nM T27812 C01QKJ 44453119 Ki = 4750 nM T27812 CB06JG 44454485 IC50 = 7500 nM T27812 CISA76 44454488 IC50 > 10000 nM T27812 CE1X7O 44454489 IC50 > 10000 nM T27812 CYRU93 44454493 IC50 = 1300 nM T27812 CKJ2D3 44454526 IC50 = 2000 nM T27812 CB9M0F 44454528 IC50 = 1700 nM T27812 CYCB65 44454556 IC50 = 3200 nM T27812 CH4JN9 44454557 IC50 = 830 nM T27812 CJB41D 44454559 IC50 > 10000 nM T27812 CQ87FZ 44454585 IC50 > 10000 nM T27812 C8LR9P 44454660 IC50 = 150 nM T27812 C3T5HK 44454663 IC50 = 77 nM T27812 C89SJY 44454690 IC50 > 10000 nM T27812 CYZ39A 44454694 IC50 > 10000 nM T27812 C0QVN8 44454719 IC50 > 10000 nM T27812 C01XOI 44454744 IC50 = 8.3 nM T27812 C1H0FI 44454746 IC50 = 3500 nM T27812 C43QBZ 44454747 IC50 = 4400 nM T27812 CEY3T6 44454767 IC50 = 100 nM T27812 C8FBC2 44454794 IC50 > 10000 nM T27812 CJBD47 44454795 IC50 = 640 nM T27812 C4WOL9 44454797 IC50 = 4800 nM T27812 CU49TR 44454860 IC50 = 1700 nM T27812 COX3W0 44454862 IC50 = 1200 nM T27812 CQF13W 44454863 IC50 = 1100 nM T27812 CU21QR 44454893 IC50 = 4400 nM T27812 CU8K7O 44454894 IC50 = 160 nM T27812 CVU57D 44454896 IC50 > 10000 nM T27812 C1P5VQ 44454931 IC50 = 1300 nM T27812 CZ2X0T 44454932 IC50 > 10000 nM T27812 CXC09Y 44454967 IC50 = 2744 nM T27812 C75SEP 44454968 IC50 = 2798 nM T27812 C5LN9M 44454971 IC50 = 1424 nM T27812 CIH52C 44455025 IC50 = 25 nM T27812 CI5T8S 44455135 IC50 = 2534 nM T27812 CGI6A7 44455136 IC50 = 3880 nM T27812 CM9OW7 44455170 IC50 = 1052 nM T27812 C8E4AF 44455171 IC50 = 3378 nM T27812 CH4N8R 44455206 IC50 = 3172 nM T27812 CEZR53 44455270 IC50 = 2686 nM T27812 CVDA26 44455301 IC50 = 1493 nM T27812 C0UC6P 44455338 IC50 = 1503 nM T27812 C89COF 44455373 IC50 > 10000 nM T27812 CRFJ58 44455391 IC50 = 6236 nM T27812 CZL97F 44455426 Ki = 3516 nM T27812 CMNX58 44455445 IC50 = 3667 nM T27812 CC09EJ 44455512 Ki = 10 nM T27812 C6YQU9 44455589 IC50 = 10 nM T27812 C9PG3H 44455590 IC50 = 16 nM T27812 C1BR2G 44455619 IC50 = 14 nM T27812 CO1X6Z 44455620 IC50 = 17 nM T27812 C8F5CI 44455622 IC50 = 7 nM T27812 C0EM9R 44455651 IC50 = 12 nM T27812 CW7E6X 44455652 IC50 = 11 nM T27812 C3W1EZ 44455653 IC50 = 28 nM T27812 CI4K0E 44455654 IC50 = 37 nM T27812 CZV45C 44455655 IC50 = 13 nM T27812 C0L9YB 44455677 IC50 = 12 nM T27812 CV10IJ 44455678 IC50 = 13 nM T27812 CK47LB 44455681 IC50 = 5 nM T27812 CIW6A1 44455707 IC50 = 73 nM T27812 CR24HA 44455708 IC50 = 22 nM T27812 COV02B 44455738 IC50 = 32 nM T27812 C3CXW8 44455739 IC50 = 6 nM T27812 CO4B1F 44455740 IC50 = 13 nM T27812 C3I6TO 44455742 IC50 = 6 nM T27812 C76JRV 44455761 IC50 = 190 nM T27812 CSX82U 44455763 IC50 = 282 nM T27812 C16SFL 44455822 Ki = 47 nM T27812 CB8AN0 44455850 Ki = 6.4 nM T27812 CEY02T 44455851 Ki = 116 nM T27812 C8MV5J 44455895 IC50 = 405 nM T27812 CAB61T 44455930 IC50 = 31 nM T27812 CD90LW 44456110 IC50 = 56 nM T27812 C2K8HO 44456196 IC50 = 106 nM T27812 CT70DM 44456231 Ki = 15 nM T27812 C08MBY 44456312 Ki = 6.3 nM T27812 CMT7G2 44456313 IC50 = 140 nM T27812 C12XGE 44456400 Ki > 10000 nM T27812 CI8HF6 44456422 IC50 = 53 nM T27812 CVTY18 44456425 IC50 = 17 nM T27812 CB68FX 44456464 IC50 = 593 nM T27812 C8TPF7 44456465 IC50 = 992 nM T27812 C6SL0P 44456466 IC50 = 2200 nM T27812 CS74YL 44457050 Ki = 498 nM T27812 C36OQY 44457051 Ki = 733 nM T27812 CKI8L5 44457058 Ki = 614 nM T27812 CQS23B 44457059 Ki = 90.88 nM T27812 CC9ZF1 44462051 Ki = 0.38 nM T27812 CN3H5R 44462082 Ki = 23 nM T27812 CL9O8M 44462783 IC50 = 11 nM T27812 C91PCM 44466344 Ki = 0.2512 nM T27812 CZA36I 44466345 Ki = 6.31 nM T27812 C63XKS 44467026 Ki = 1.585 nM T27812 CH4WM3 44467027 Ki = 1.259 nM T27812 C3T4BX 44467028 Ki = 3.981 nM T27812 CG4R7A 44467101 Ki = 1.995 nM T27812 CW2K9E 44467103 Ki = 3.981 nM T27812 CL0JR9 44467104 Ki = 2.512 nM T27812 C4CX9E 44467173 Ki = 39.81 nM T27812 CG4H1R 44467174 Ki = 39.81 nM T27812 CLU6A0 44467177 Ki = 3.981 nM T27812 C4RBV8 44467889 Ki = 1.259 nM T27812 CJB37C 44467892 Ki = 6.31 nM T27812 CF4ZM8 44467957 Ki = 0.7943 nM T27812 CTO9R8 44467960 Ki = 12.59 nM T27812 C4DL5C 44469677 IC50 > 10000 nM T27812 C2QK4J 44472590 IC50 = 1613 nM T27812 CQ8C3F 44472591 IC50 = 200 nM T27812 CC2TA5 44472592 IC50 = 700 nM T27812 CWN95E 44472610 IC50 = 4400 nM T27812 C1H2ZT 44472612 IC50 = 2500 nM T27812 C9G5ID 44472613 IC50 = 1100 nM T27812 C5N4KE 44472633 IC50 = 7100 nM T27812 CM6Q7W 44474580 Ki = 7.47 nM T27812 C73XSD 44474582 Ki = 30.4 nM T27812 C68VDK 44474583 Ki = 33.2 nM T27812 C21WPR 44474586 Ki = 2.01 nM T27812 C8UON6 44474625 IC50 > 10000 nM T27812 C6HVU1 44474629 IC50 > 10000 nM T27812 C3DHG0 44511399 IC50 = 181 nM T27812 C68NXC 44517723 IC50 = 4800 nM T27812 CU9MO1 44539110 Ki = 0.07943 nM T27812 CAL8V3 44539203 Ki = 15.85 nM T27812 CO1E5C 44539964 IC50 = 32 nM T27812 CLMY52 44539967 IC50 = 143 nM T27812 CLO73R 44540428 IC50 = 138 nM T27812 CV92IJ 44541354 IC50 = 0.068 nM T27812 C5Q3NI 44542504 IC50 > 100 nM T27812 C5F1UC 44542505 Ki > 10000 nM T27812 CYX7H5 44542510 IC50 = 400 nM T27812 C71QGD 44542511 IC50 > 100 nM T27812 C8V7UL 44542657 Ki = 6200 nM T27812 C6ECJ1 44542658 IC50 = 185 nM T27812 C2EDU6 44542955 IC50 > 100 nM T27812 CTW5I9 44542956 Ki > 10000 nM T27812 C03MXJ 44543264 IC50 > 100 nM T27812 CL5UK7 44543265 IC50 = 473 nM T27812 CBL30Z 44543269 Ki = 6200 nM T27812 CHIY92 44543270 Ki > 10000 nM T27812 C1YIC9 44560434 Ki = 660 nM T27812 C7G9WM 44560436 Ki > 2000 nM T27812 C35XEU 44560438 Ki > 2000 nM T27812 CBTX17 44560440 Ki > 2000 nM T27812 CB0K6T 44560442 Ki = 908 nM T27812 CWCT08 44560444 Ki > 2000 nM T27812 C69ETG 44560446 Ki = 387 nM T27812 CK2PD5 44560493 Ki = 522 nM T27812 C2SZ1B 44560495 Ki > 2000 nM T27812 C9U5SE 44560498 Ki = 366 nM T27812 CNK4F6 44560500 Ki = 864 nM T27812 CU05HZ 44560502 Ki = 297 nM T27812 C87VZD 44560504 Ki = 1000 nM T27812 CV0BF4 44560506 Ki = 1800 nM T27812 CS9N0U 44560575 IC50 = 320 nM T27812 CYNS29 44560577 IC50 > 10000 nM T27812 CF5BX9 44560599 Ki > 2000 nM T27812 CNF81T 44560602 Ki = 72 nM T27812 CWB6S3 44560604 Ki = 113 nM T27812 CJQ4R5 44560606 Ki = 79 nM T27812 C7TO9F 44560608 Ki = 85 nM T27812 C17ZEN 44560622 IC50 = 2000 nM T27812 CN1K6R 44560623 IC50 = 9000 nM T27812 C9BV0O 44560624 IC50 = 50 nM T27812 CY72NM 44560625 IC50 = 130 nM T27812 C0FW5J 44560626 IC50 = 1400 nM T27812 CLW2R6 44560627 IC50 = 300 nM T27812 CI1XD4 44560628 IC50 = 3500 nM T27812 C1NCT4 44560653 Ki = 42.9 nM T27812 C8MPN0 44560655 Ki = 89.7 nM T27812 CWG57V 44560657 Ki = 14.4 nM T27812 CH79ZT 44560659 Ki = 41.1 nM T27812 C51DKQ 44560671 IC50 = 8000 nM T27812 CBMT59 44560672 IC50 = 3000 nM T27812 C1R8PQ 44560673 IC50 > 10000 nM T27812 CGK29S 44560675 IC50 = 370 nM T27812 CG4YN5 44560676 IC50 = 150 nM T27812 CNM1Q6 44560708 IC50 = 700 nM T27812 CG6FL1 44560709 IC50 = 3300 nM T27812 CL9J2E 44560710 IC50 = 3000 nM T27812 C36IOW 44560711 IC50 = 1100 nM T27812 CLM2F8 44560712 IC50 = 2300 nM T27812 C3OG8F 44560713 IC50 = 5000 nM T27812 C9B5CE 44560714 IC50 > 10000 nM T27812 CR8OX1 44562611 IC50 = 4.27 nM T27812 CL64BM 44562612 IC50 = 77.5 nM T27812 CVB0Q6 44562613 IC50 = 31.2 nM T27812 C02CWF 44562614 IC50 = 25.4 nM T27812 C7CSF8 44562615 IC50 = 9.71 nM T27812 CNJM41 44562616 IC50 = 88 nM T27812 CP7RQ8 44562623 IC50 = 4000 nM T27812 CHE68Z 44562624 IC50 = 3000 nM T27812 CR4TG7 44562625 IC50 = 700 nM T27812 CH32FI 44562626 IC50 = 700 nM T27812 CX1P3L 44562627 IC50 = 2200 nM T27812 C0S8ZG 44562682 IC50 = 500 nM T27812 C2HKE0 44562772 IC50 = 1800 nM T27812 C50WKO 44562773 IC50 = 50 nM T27812 C3JD7Y 44562774 IC50 = 5 nM T27812 CS0LD7 44562775 IC50 = 36 nM T27812 C7AC8Z 44562776 IC50 = 6 nM T27812 CU6G4W 44562777 IC50 = 200 nM T27812 CCA0H2 44562815 IC50 = 150 nM T27812 CQ0I5R 44562816 IC50 = 100 nM T27812 CC1IF3 44562817 IC50 = 14 nM T27812 C3VP6N 44562943 IC50 = 4.67 nM T27812 C7DS0M 44562944 IC50 = 74.7 nM T27812 C4XL2E 44562989 IC50 = 4.02 nM T27812 C4UG5R 44562990 IC50 = 2.43 nM T27812 CY84FH 44563029 IC50 = 3.46 nM T27812 C5N9FG 44563030 IC50 = 34.4 nM T27812 C5J6HU 44563054 IC50 = 36 nM T27812 C6B2FI 44563127 IC50 = 9.35 nM T27812 CL0DS9 44563128 IC50 = 3.78 nM T27812 C0J2GS 44563163 IC50 = 4.37 nM T27812 C67TOD 44563164 IC50 = 61.2 nM T27812 CL5HW8 44563165 IC50 = 39.6 nM T27812 C7BRD0 44563202 IC50 = 28.9 nM T27812 CDX3R8 44563203 IC50 = 41.2 nM T27812 C5QX2S 44563204 IC50 = 31.1 nM T27812 CF4ZK8 44563205 IC50 = 17 nM T27812 C3ZUH6 44563206 IC50 = 20.7 nM T27812 CR28PD 44563213 IC50 = 10 nM T27812 CU4PD5 44563214 IC50 = 184 nM T27812 CJ9O6U 44563238 IC50 = 9.2 nM T27812 CB8P3I 44563239 IC50 = 187 nM T27812 CB9NG8 44563240 IC50 = 115 nM T27812 CN5U4V 44563241 IC50 = 9.81 nM T27812 CLJ7C2 44563242 IC50 = 5.73 nM T27812 C2OX9D 44563243 IC50 = 7.49 nM T27812 C1VQ5X 44563244 IC50 = 4.19 nM T27812 CGKL94 44563257 IC50 = 1400 nM T27812 C8TYL3 44563258 IC50 = 2500 nM T27812 C8XUD6 44563259 IC50 > 10000 nM T27812 CIG6Z4 44563260 IC50 = 5700 nM T27812 C9VFW6 44563261 IC50 = 3500 nM T27812 C9N0RT 44563646 Ki = 0.43 nM T27812 CEG7S1 44563647 Ki = 0.33 nM T27812 C41KWG 44563667 Ki = 0.26 nM T27812 CI6A1Q 44563668 Ki = 0.33 nM T27812 CL83PU 44563669 Ki = 15.2 nM T27812 CJD73U 44565305 IC50 = 194 nM T27812 CM8LR1 44568174 IC50 = 3 nM T27812 CCRI61 44568175 IC50 = 25 nM T27812 CB3VF8 44568176 IC50 = 30 nM T27812 C6T2BK 44568293 IC50 = 17 nM T27812 CA1NJ9 44568294 IC50 = 660 nM T27812 CA21KI 44568295 IC50 = 4 nM T27812 CX50DP 44568296 IC50 = 4 nM T27812 COB14G 44568297 IC50 = 3 nM T27812 C3I6FM 44568320 IC50 = 6 nM T27812 C4QYH2 44568321 IC50 = 60 nM T27812 CKT30F 44568322 IC50 = 26 nM T27812 C1HA7U 44568323 IC50 = 30 nM T27812 C9CJP2 44568324 IC50 = 1900 nM T27812 C81XJM 44568325 IC50 = 3 nM T27812 CFE30X 44568348 IC50 = 20 nM T27812 C3SW7N 44568349 IC50 = 10 nM T27812 CLTG36 44568350 IC50 = 3 nM T27812 C9MNC0 44568351 IC50 = 5 nM T27812 CB58VS 44568378 IC50 = 10 nM T27812 CYN68I 44568379 IC50 = 100 nM T27812 CY3NQ8 44568652 IC50 = 30 nM T27812 C02GHU 44568653 IC50 = 5 nM T27812 CAO2I3 44568689 IC50 = 40 nM T27812 CM1SR3 44568690 IC50 > 1000 nM T27812 C8HNK7 44568691 IC50 = 50 nM T27812 C3HQ2F 44568692 IC50 = 45 nM T27812 C7FBU8 44568693 IC50 = 4 nM T27812 CD48SQ 44568694 IC50 = 5 nM T27812 CSZ7V2 44568750 IC50 = 70 nM T27812 CWG32I 44572166 Ki = 1042 nM T27812 C97VKX 44572751 Ki = 3824 nM T27812 CJ1VI8 44572802 Ki = 5441 nM T27812 CU25XD 44572810 Ki = 2710 nM T27812 CO1VA0 44574739 IC50 = 33 nM T27812 CIUN13 44574783 IC50 = 2105 nM T27812 CO40XG 44574784 IC50 = 836 nM T27812 CX15IN 44574883 IC50 = 439 nM T27812 CX07AK 44574884 IC50 = 416 nM T27812 C6S4IO 44576826 Ki = 39 nM T27812 C7WO9Z 44576828 Ki = 7 nM T27812 CE5JC1 44576830 Ki = 252 nM T27812 C4XBZ0 44576832 Ki = 76 nM T27812 COT0K9 44576862 Ki = 54 nM T27812 CYXV83 44576864 Ki = 18 nM T27812 CS4XT1 44576866 Ki = 730 nM T27812 CCB06N 44576868 Ki = 81 nM T27812 CV45DH 44576870 Ki = 620 nM T27812 C42FLK 44576888 Ki = 19 nM T27812 COP7S3 44576890 Ki = 138 nM T27812 C4ISW9 44576892 Ki = 161 nM T27812 CC2GJ8 44578041 IC50 = 41 nM T27812 CS71BE 44578042 IC50 = 195 nM T27812 CHE5X2 44578075 IC50 = 26 nM T27812 C32VHN 44578076 IC50 = 123 nM T27812 CL2MG7 44578077 IC50 = 91 nM T27812 C4T5JW 44578112 IC50 = 24 nM T27812 CEO36B 44578113 IC50 > 400 nM T27812 CC0A8W 44578263 Ki = 544 nM T27812 CFJB16 44578266 Ki = 4120 nM T27812 CE54ZK 44578267 Ki = 5620 nM T27812 CSFE81 44578268 Ki = 5680 nM T27812 CAQK40 44578269 Ki > 10000 nM T27812 C5P0QK 44578270 Ki > 10000 nM T27812 CQ30GC 44578271 Ki = 410 nM T27812 C8HB0Z 44578272 Ki = 5350 nM T27812 CV63SW 44578313 Ki = 50 nM T27812 CH3U5D 44578314 Ki = 4690 nM T27812 C8XAO4 44578315 Ki = 5280 nM T27812 CS70JE 44578316 Ki = 2890 nM T27812 CAP14F 44578317 Ki = 1250 nM T27812 CUVQ89 44578318 Ki = 2700 nM T27812 C17YVO 44578319 Ki = 3330 nM T27812 CPQC54 44578368 Ki = 869 nM T27812 CA5I3W 44578369 Ki = 5810 nM T27812 CTE6V8 44578370 Ki = 787 nM T27812 C4VO1L 44578371 Ki = 764 nM T27812 CXZ05B 44578372 Ki = 427 nM T27812 CVXD80 44578373 Ki = 353 nM T27812 C8AP4K 44578374 Ki = 444 nM T27812 CDMH40 44578375 Ki = 5010 nM T27812 CAVH68 44578853 Ki > 1000 nM T27812 C16GJP 44578854 Ki > 1000 nM T27812 CW9FQ8 44578855 Ki = 3464 nM T27812 C2H8IL 44578856 Ki = 5977 nM T27812 CI2R0O 44578902 Ki > 1000 nM T27812 CVG6E5 44579403 IC50 = 600 nM T27812 C5JOP4 44579404 IC50 = 750 nM T27812 CY01LU 44579444 IC50 = 5 nM T27812 C4H3AR 44579445 IC50 = 10 nM T27812 C4DZI3 44579446 IC50 = 16 nM T27812 C5KQH6 44579463 Ki > 10000 nM T27812 CJ1WX8 44579464 Ki = 230 nM T27812 C3PQ6R 44579486 IC50 = 7 nM T27812 C7ZXQ1 44579536 Ki = 639 nM T27812 C01PQB 44579537 Ki = 1040 nM T27812 CNZ59J 44579538 Ki = 109 nM T27812 CY65RZ 44579539 Ki > 10000 nM T27812 C0M9NK 44579564 IC50 = 9 nM T27812 CUQV50 44579565 IC50 > 1000 nM T27812 C1MQ2P 44579566 IC50 = 5 nM T27812 C18FPJ 44579567 IC50 > 1000 nM T27812 CN9Y6Q 44579595 Ki > 10000 nM T27812 C2VS4Z 44579596 Ki > 10000 nM T27812 CV9NK7 44579597 Ki = 177 nM T27812 C6E8LD 44579598 Ki > 1000 nM T27812 CS91HK 44579613 IC50 > 10000 nM T27812 CZO5Y8 44580740 Ki = 0.3981 nM T27812 C4N6PM 44580741 Ki = 0.7943 nM T27812 C0XVL5 44580783 Ki = 3.981 nM T27812 C4SD7P 44580784 Ki = 3.981 nM T27812 CRCH48 44582675 Ki = 2207 nM T27812 CEJ4R8 44582676 Ki = 3087 nM T27812 C5QB4K 44582678 Ki = 2646 nM T27812 C01RCI 44582705 Ki = 1009 nM T27812 C3L5ER 44583033 IC50 = 0.061 nM T27812 CBIO97 44585469 IC50 = 0.05 ug.mL-1 T27812 C4HJE6 44586246 Ki = 6.46 nM T27812 CXKQ61 44587384 IC50 = 1100 nM T27812 CZLV68 44587385 IC50 = 3100 nM T27812 C8SFJ1 44587386 IC50 = 10000 nM T27812 CPBR52 44587387 IC50 = 3500 nM T27812 C4D7GP 44587388 IC50 > 10000 nM T27812 CRL0H9 44587389 IC50 = 640 nM T27812 C5PV7Q 44587390 IC50 = 6000 nM T27812 C5IUL8 44587443 IC50 = 7800 nM T27812 C59KDV 44587445 IC50 > 10000 nM T27812 CLCE75 44587446 IC50 > 10000 nM T27812 CPF01B 44587447 IC50 = 3000 nM T27812 CIL89C 44587448 IC50 = 4500 nM T27812 CF0I6D 44587449 IC50 = 6700 nM T27812 C0J4LS 44587450 IC50 = 390 nM T27812 CZVX16 44587463 IC50 = 6500 nM T27812 C6UI9D 44587464 IC50 = 230 nM T27812 C6YQS2 44587465 IC50 = 140 nM T27812 CNV4I9 44587466 IC50 = 1500 nM T27812 CL10BT 44587467 IC50 = 90 nM T27812 CX5KZ1 44587468 IC50 = 3600 nM T27812 C0OYJ4 44587469 IC50 = 2700 nM T27812 C2HUA1 44587470 IC50 = 2700 nM T27812 CIW41M 44587471 IC50 = 3100 nM T27812 CCKE83 44587472 IC50 = 4500 nM T27812 C4SGR3 44587473 IC50 = 3000 nM T27812 C47OBV 44587474 IC50 > 10000 nM T27812 CQ79SU 44587475 IC50 = 100 nM T27812 CUE9C6 44587476 IC50 = 150 nM T27812 C37ZEB 44587477 IC50 = 4000 nM T27812 CY0F1M 44587482 IC50 = 4000 nM T27812 CL5M2J 44587483 IC50 = 2800 nM T27812 CRN0Z1 44587484 IC50 = 2700 nM T27812 CTN0Q1 44587485 IC50 = 4600 nM T27812 CAHW83 44587486 IC50 > 10000 nM T27812 CJY60H 44587487 IC50 = 3200 nM T27812 C3OL1M 44587488 IC50 = 300 nM T27812 C56QTZ 44587489 IC50 = 35 nM T27812 CD60KY 44587995 Ki = 1.7 nM T27812 CZ98JO 44587997 Ki = 4.8 nM T27812 CAXU48 44587999 Ki = 3.1 nM T27812 C6FPZ9 44588001 Ki = 2.9 nM T27812 C8F7IT 44588013 Ki = 3.5 nM T27812 C8LUE2 44588015 Ki = 7.5 nM T27812 C7Y4QV 44588017 Ki = 135 nM T27812 C5JQY4 44588019 Ki = 29 nM T27812 C62JSH 44588021 Ki = 100 nM T27812 C43ODT 44588187 Ki = 0.95 nM T27812 CKPE78 44588189 Ki = 4.3 nM T27812 C57QYV 44588191 Ki = 2.9 nM T27812 CPR9K4 44588193 Ki = 8.3 nM T27812 CLIV63 44588195 Ki = 5.5 nM T27812 CN6RC7 44588197 Ki = 4.1 nM T27812 CH18RV 44588223 Ki = 2 nM T27812 CXA2D6 44588225 Ki = 3.5 nM T27812 C4RZ1U 44588227 Ki = 1 nM T27812 CQSC48 44588229 Ki = 860 nM T27812 C60NYB 44588704 IC50 = 109 nM T27812 CB27TM 44589076 IC50 = 146 nM T27812 C4WB1N 44589201 Ki = 23 nM T27812 C69KAB 44590643 IC50 = 2071 nM T27812 CLQ2N4 44590644 IC50 = 1117 nM T27812 CJ2D4T 44590690 IC50 = 122 nM T27812 C0RHT8 44590691 Ki = 20 nM T27812 CQCG57 44590692 IC50 = 2.5 nM T27812 CS7H9U 44590693 IC50 = 11.7 nM T27812 C38PUH 44590694 Ki = 2.1 nM T27812 CDB8Z5 44590725 IC50 = 17.5 nM T27812 C0N5RO 44590726 Ki = 0.8 nM T27812 C4H6PT 44590727 IC50 = 2.6 nM T27812 C3TUD7 44590728 Ki = 4 nM T27812 CNL38Q 44590729 Ki = 2 nM T27812 C7RBE8 44590819 Ki = 92 nM T27812 CYBL93 44590820 Ki = 86 nM T27812 CI6R1Z 44592120 IC50 = 3 nM T27812 C1QO8J 44592121 IC50 = 4 nM T27812 C7LKH8 44592122 IC50 > 400 nM T27812 CVT6R5 44592123 IC50 = 14 nM T27812 C04UVE 44592152 IC50 = 138 nM T27812 C4KM6A 44592153 IC50 = 30 nM T27812 C12UEV 44592154 IC50 > 400 nM T27812 CV8E7O 44592155 IC50 = 16 nM T27812 CK47SV 44592156 IC50 = 119 nM T27812 C4W1XJ 44592157 IC50 = 5 nM T27812 CMS5I2 44592158 IC50 = 13 nM T27812 CSU06J 44592195 IC50 = 0.3 nM T27812 CZ6L3I 44592196 IC50 = 2 nM T27812 C4EH6O 44592207 Ki = 100 nM T27812 CZ5I1N 44592208 Ki = 158.49 nM T27812 CKM8T7 44592209 Ki = 19.95 nM T27812 CC52XI 44592242 IC50 = 5 nM T27812 CJO9K5 44592245 IC50 = 4 nM T27812 CDJ32U 44592249 Ki = 158.49 nM T27812 CS2FL4 44592250 Ki = 125.89 nM T27812 CL17WU 44592251 Ki = 199.53 nM T27812 CJCL64 44592252 Ki = 63.1 nM T27812 CM0I3E 44592294 Ki = 5.012 nM T27812 CQ04EG 44592295 Ki = 12.59 nM T27812 C65XQL 44592296 Ki = 7.943 nM T27812 CEB2S1 44592297 Ki = 1.995 nM T27812 CP51QS 44592332 Ki = 0.3981 nM T27812 CD2Z4J 44592333 Ki = 0.5012 nM T27812 C7NCT2 44592334 Ki = 0.3162 nM T27812 CHY20X 44592335 Ki = 0.7943 nM T27812 C5H7XK 44592371 Ki = 39.81 nM T27812 CQ12YR 44593444 IC50 = 0.35 nM T27812 CPH6S0 44593451 IC50 = 1400 nM T27812 C30HFZ 44593522 IC50 = 10 nM T27812 CI3T5N 44593629 Ki = 120 nM T27812 C1DI5Z 44593686 IC50 = 1600 nM T27812 C7YLS4 44593687 IC50 = 1300 nM T27812 C6KGF2 44593688 IC50 = 2600 nM T27812 CU8F9L 44593689 IC50 = 1200 nM T27812 CR18ZA 44593690 IC50 = 5600 nM T27812 C20YZD 44593691 IC50 = 6000 nM T27812 CN52LH 44593692 IC50 = 500 nM T27812 C7IU8S 44593694 IC50 = 900 nM T27812 C9SM4D 44593695 IC50 = 960 nM T27812 CSQ14O 44593696 IC50 = 560 nM T27812 CHD0R7 44593712 IC50 = 10.1 nM T27812 CPK6N9 44593714 IC50 = 71.6 nM T27812 C5HSO3 44593715 IC50 = 291 nM T27812 CAXK49 44593716 IC50 > 1000 nM T27812 C4WBK1 44593717 IC50 > 1000 nM T27812 CI10GR 44610722 IC50 = 4.6 nM T27812 CW84TH 44610723 IC50 = 3.5 nM T27812 CPIB93 44610724 IC50 = 3.5 nM T27812 CINL72 44613065 EC50 = 25118.86 nM T27812 C70ASV 44613066 EC50 = 19498.45 nM T27812 CYQ08F 44613069 EC50 = 12882.5 nM T27812 C8LE4X 44613187 EC50 = 20892.96 nM T27812 CCF91E 44613190 EC50 = 29512.09 nM T27812 CN61TV 44613191 EC50 = 2454708.92 nM T27812 CJ1Z2G 44613327 EC50 = 3981.07 nM T27812 CS7JI9 44613328 EC50 = 8128.31 nM T27812 CC1O6A 44613454 EC50 = 18620.87 nM T27812 CZ2P0I 44613457 EC50 > 100000 nM T27812 CSQ65B 44613459 EC50 = 44668.36 nM T27812 CM7I0R 44613581 EC50 = 19142.56 nM T27812 CN1G4T 44613689 EC50 = 14454.4 nM T27812 CP4D9B 44613813 EC50 = 2570.4 nM T27812 C3CA7P 44613814 EC50 = 1949844.6 nM T27812 CVR29I 44625567 IC50 = 12.59 nM T27812 C24WVM 44625568 IC50 = 7.943 nM T27812 COM81X 44625569 IC50 = 1 nM T27812 CR8I3P 44625570 IC50 = 7.943 nM T27812 C2D0TJ 44625571 IC50 = 0.7943 nM T27812 C6LD5P 44625653 IC50 = 100 nM T27812 CU3LE6 44626329 Ki = 22 nM T27812 C0A3WN 44626374 IC50 = 343 nM T27812 CY47CM 45101948 IC50 = 427 nM T27812 CND19I 45102009 IC50 = 265 nM T27812 CW0RU3 45102635 Ki > 4900 nM T27812 C0DLU3 45109862 IC50 = 137 nM T27812 CR83KY 45139778 IC50 = 29 nM T27812 CB16EP 45139780 IC50 = 21 nM T27812 C15AOE 45139782 IC50 = 84 nM T27812 CBDG89 45139784 IC50 = 499 nM T27812 C6ZL5S 45139960 IC50 = 1123 nM T27812 CAKF28 45139962 IC50 = 5.5 nM T27812 C2RH4W 45139964 IC50 = 2.8 nM T27812 C10AOU 45139966 IC50 = 813 nM T27812 C1AWI8 45139968 IC50 = 280 nM T27812 CSC30M 45139970 IC50 = 4519 nM T27812 CEB8M7 45139972 IC50 = 8971 nM T27812 CHRV87 45140168 IC50 = 1969 nM T27812 CO03PE 45140170 IC50 = 4917 nM T27812 CO1KI6 45140172 IC50 = 2871 nM T27812 C1S5GM 45140174 IC50 = 5293 nM T27812 CXJ80R 45140176 IC50 = 364 nM T27812 CRW5G7 45140178 IC50 = 4992 nM T27812 CXJ6A2 45140180 IC50 = 1099 nM T27812 CT6XO9 45140370 IC50 = 1614 nM T27812 CUOD26 45140371 IC50 = 194 nM T27812 C7MB5N 45141377 IC50 > 100 nM T27812 CMSH89 45141378 IC50 > 100 nM T27812 C05NYK 45141587 IC50 = 154 nM T27812 CTL0U6 45141609 IC50 > 100 nM T27812 CB9QZ6 45263405 IC50 = 3.9 nM T27812 CP3S0Q 45266826 EC50 = 118 nM T27812 CPGO97 45267145 IC50 = 5 nM T27812 CTL3Z5 45267156 IC50 = 7 nM T27812 CT15YP 45267165 IC50 = 10 nM T27812 CZ3DW4 45267166 IC50 = 11 nM T27812 C5DGO1 45267167 IC50 = 8 nM T27812 CP7XE6 45267597 Ki = 210 nM T27812 CK58HY 45267611 Ki = 661 nM T27812 C3D9TN 45267621 Ki = 1000 nM T27812 CV1W8D 45267665 IC50 = 126 nM T27812 CEWR12 45268018 IC50 = 3 nM T27812 CD8G9N 45268026 IC50 = 7 nM T27812 C9VB2Y 45268114 IC50 = 2.6 nM T27812 C4DZO1 45268459 IC50 = 17 nM T27812 CRP90V 45268466 Ki = 237 nM T27812 CSJ4L2 45268478 Ki = 113 nM T27812 C9IJK8 45268483 IC50 > 10000 nM T27812 CQJ9X1 45268495 Ki = 6.31 nM T27812 CO2X9T 45268882 IC50 = 95 nM T27812 C71XIB 45268898 IC50 = 3 nM T27812 CHP12M 45268914 IC50 = 3 nM T27812 CUQ23Z 45268922 IC50 = 36 nM T27812 CZC09M 45269305 IC50 = 14 nM T27812 CFJ17A 45269306 IC50 = 11 nM T27812 CNA70T 45269316 IC50 = 17 nM T27812 C1SB8A 45269317 IC50 = 38 nM T27812 C5OED7 45269318 Ki = 39 nM T27812 CF2P9H 45269325 Ki = 62 nM T27812 CQ03ZU 45269337 Ki = 581 nM T27812 CXE36D 45269351 Ki = 187 nM T27812 CVA9E0 45269726 IC50 = 80 nM T27812 CS0Z8C 45269735 IC50 = 76 nM T27812 CL6W3X 45269754 IC50 = 8 nM T27812 CDM73H 45270136 IC50 = 8 nM T27812 CX31KD 45270149 Ki = 654 nM T27812 C3GA6N 45270158 Ki = 857 nM T27812 C3KI7Q 45270163 Ki = 457 nM T27812 C0QR1E 45270171 Ki = 2870 nM T27812 C6YI5N 45270172 Ki = 663 nM T27812 CZ9DA3 45270173 Ki = 330 nM T27812 C2M8FY 45270563 IC50 = 7 nM T27812 C13GPD 45270570 IC50 = 5 nM T27812 CM48NS 45270571 IC50 = 10 nM T27812 CH32XG 45270576 IC50 > 400 nM T27812 C0HV4C 45270577 IC50 = 6 nM T27812 COFD89 45270589 IC50 = 16 nM T27812 CEX26T 45270595 IC50 = 8 nM T27812 CZ9OC8 45270973 IC50 = 15 nM T27812 C13QSU 45270993 Ki = 348 nM T27812 CU9HV3 45271001 Ki = 802 nM T27812 CBW87K 45271004 IC50 = 59 nM T27812 C71AON 45271011 Ki = 776 nM T27812 CI01KJ 45271024 Ki = 25.12 nM T27812 C62UVG 45271383 IC50 = 61 nM T27812 C61TGI 45271390 IC50 = 3 nM T27812 CE8Z1K 45271821 IC50 = 14 nM T27812 CLD3T9 45271838 IC50 = 24 nM T27812 C1S6TI 45271840 Ki = 118 nM T27812 C3QAP5 45271853 Ki = 1090 nM T27812 CP7K0V 45271861 IC50 = 130 nM T27812 CFG5Z3 45271864 Ki = 5210 nM T27812 C3AJ7I 45271873 Ki = 398.11 nM T27812 CT04SP 45271883 Ki = 19.95 nM T27812 C1MKJ3 45272270 IC50 = 77 nM T27812 C1G9IK 45272302 IC50 = 17 nM T27812 C5DE4U 45272692 IC50 = 17 nM T27812 CPM1U3 45272720 Ki = 64 nM T27812 C4VAE9 45272734 Ki = 587 nM T27812 C4P1FO 45273132 IC50 = 9 nM T27812 CUK91L 45273154 IC50 = 14 nM T27812 C5LB6F 45273161 IC50 = 16 nM T27812 C2DB0Y 45273169 IC50 = 7 nM T27812 C6KGT7 45273264 IC50 = 1.1 nM T27812 C1JLQ3 45273630 IC50 = 26 nM T27812 C7HQ9B 45273656 IC50 = 76 nM T27812 CT3V0B 45273663 Ki = 109 nM T27812 CINR73 45273666 Ki = 1080 nM T27812 C3Q0GZ 45273673 Ki = 1990 nM T27812 CZU06K 45273676 Ki = 31.62 nM T27812 C2J0GO 45278647 IC50 = 7 nM T27812 C7X3LG 45278648 IC50 = 133 nM T27812 CG64BP 45278720 IC50 = 11.1 nM T27812 CD9HF8 45278721 IC50 = 11.8 nM T27812 CYT87H 45278722 IC50 = 25.8 nM T27812 C8QK9C 45278723 IC50 = 35.9 nM T27812 C2M5HA 45278725 IC50 = 93 nM T27812 CXJ8L6 45278729 IC50 = 85 nM T27812 CAQ40Z 45278802 IC50 = 76 nM T27812 CARO27 45278803 IC50 = 110 nM T27812 CFG01K 45278804 IC50 = 92 nM T27812 CZ71RN 45278805 IC50 = 61.7 nM T27812 CFN4D9 45278806 IC50 = 182 nM T27812 CZN6M7 45278882 IC50 = 420 nM T27812 C6NT3Q 45278883 IC50 = 298 nM T27812 CA58GM 45278884 IC50 = 80.2 nM T27812 C21JKF 45278885 IC50 = 53.6 nM T27812 CS5BA4 45278886 IC50 = 266 nM T27812 C4TXE8 45278964 IC50 = 235 nM T27812 CPI26X 45278965 IC50 = 14.3 nM T27812 C1NR0P 45278966 IC50 = 125 nM T27812 CYK65H 45278967 IC50 = 213 nM T27812 C0EGV6 45278968 IC50 = 352 nM T27812 CWI2S0 45279043 IC50 = 412 nM T27812 CN7V2L 45279044 IC50 = 92 nM T27812 C2AW3R 45279045 IC50 = 77 nM T27812 CF7O1A 45279046 IC50 = 110 nM T27812 CM46OZ 45279047 IC50 = 350 nM T27812 CB02TI 45279127 IC50 = 381 nM T27812 CS62HT 45279130 IC50 = 102 nM T27812 CRM38P 45279134 IC50 = 76 nM T27812 CEZ53Y 45279210 IC50 = 76 nM T27812 CPX18C 45279212 IC50 = 149 nM T27812 CJ0X2R 45279214 IC50 = 93 nM T27812 C3NW0C 45279216 IC50 = 98 nM T27812 CX73IH 45279218 IC50 = 87 nM T27812 CGNC19 45279298 IC50 = 32 nM T27812 C8CPD7 45279300 IC50 = 21 nM T27812 CP4GI2 45279384 IC50 = 19 nM T27812 CX2ND5 45279386 IC50 = 56 nM T27812 CX5ST2 45279664 IC50 = 129 nM T27812 CKQ7S3 45279666 IC50 = 733 nM T27812 C91IRB 45279668 IC50 = 93 nM T27812 C12WRL 45279755 IC50 = 629 nM T27812 C3SUQ1 45279757 IC50 = 131 nM T27812 C63LSI 45279759 IC50 = 1159 nM T27812 CQS5X0 45378248 Ki = 0.7943 nM T27812 C7C9HW 45378386 Ki = 0.3162 nM T27812 C51WBF 45378387 Ki = 0.1995 nM T27812 CS04YD 45379827 Ki = 15.49 nM T27812 CMU6Z8 45379828 Ki = 0.7413 nM T27812 C1SCJ9 45379829 Ki = 72.44 nM T27812 CK6L2S 45379946 Ki = 0.955 nM T27812 CNQT48 45379947 Ki = 0.3162 nM T27812 C5TQ8X 45379948 Ki = 31.62 nM T27812 CP82MH 45379949 Ki = 0.5012 nM T27812 CNSK69 45379950 Ki = 1.259 nM T27812 CM61UN 45380063 Ki = 25.12 nM T27812 C97ZQE 45380064 Ki = 7.943 nM T27812 CEFO86 45380065 Ki = 1 nM T27812 C53JYC 45380066 Ki = 1.259 nM T27812 C46FLB 45380180 Ki = 3.981 nM T27812 C89XTJ 45380181 Ki = 0.3981 nM T27812 CYAE52 45380182 Ki = 25.12 nM T27812 C6BLR9 45380183 Ki = 1 nM T27812 CO8Z1P 45380184 Ki = 0.1585 nM T27812 CE1M3S 45380185 Ki = 2.512 nM T27812 C1OK5Z 45481773 Ki = 4.3 nM T27812 CS0W9K 45481774 Ki = 208 nM T27812 C5SN4D 45481775 Ki = 0.19 nM T27812 CZ02KA 45481776 Ki = 1.26 nM T27812 CCOL45 45481778 Ki = 3 nM T27812 CX68LG 45481779 Ki = 27 nM T27812 C52FTP 45481780 Ki = 5.5 nM T27812 C0NAE6 45481784 Ki = 47 nM T27812 CG75XM 45481786 Ki = 5.7 nM T27812 C5F8QK 45481787 Ki = 0.7 nM T27812 CQ89WZ 45481788 Ki = 49 nM T27812 C7BQX4 45481789 Ki = 4.5 nM T27812 C1O8ZD 45481790 Ki = 23 nM T27812 CO1Z4X 45481791 Ki = 8 nM T27812 CF6R7M 45481792 Ki = 0.6 nM T27812 CWEK71 45481794 Ki = 3.2 nM T27812 C6SN1T 45483060 IC50 = 882 nM T27812 CJOP63 45483061 IC50 = 547 nM T27812 CMH54N 45483062 IC50 = 48 nM T27812 C6BP3U 45483063 IC50 = 228 nM T27812 COT26E 45483068 IC50 = 2184 nM T27812 CDL5N0 45483069 IC50 = 48 nM T27812 C1OP5G 45483079 IC50 = 527 nM T27812 CQ4ZM0 45483080 IC50 = 417 nM T27812 C86FAI 45483083 IC50 = 1333 nM T27812 C52YIE 45483084 IC50 = 78 nM T27812 CN50YU 45483087 IC50 = 748 nM T27812 CVL4X1 45483088 IC50 = 473 nM T27812 C5DZ3N 45483089 IC50 = 626 nM T27812 CY6Z9V 45483094 IC50 = 834 nM T27812 C8AY7V 45483095 IC50 = 441 nM T27812 CVY9K0 45483096 IC50 = 1366 nM T27812 CZF8E4 45483097 IC50 = 266 nM T27812 CP7XI1 45483098 IC50 = 175 nM T27812 CQG68O 45483099 IC50 = 207 nM T27812 CS30CZ 45483103 IC50 = 221 nM T27812 C2S0EY 45483104 IC50 = 52 nM T27812 CCV7P6 45483105 IC50 = 1003 nM T27812 CCF53Z 45483112 IC50 = 377 nM T27812 C4R6AY 45483113 IC50 = 113 nM T27812 CX3HT0 45483114 IC50 = 491 nM T27812 CYWX25 45483119 IC50 = 398 nM T27812 CCFO37 45483120 IC50 = 79 nM T27812 CRZ8V3 45483130 IC50 = 865 nM T27812 C97JBX 45483401 Ki = 260 nM T27812 C9K4XC 45483416 Ki = 2 nM T27812 CZQ6H8 45483429 Ki = 40 nM T27812 C3HAF8 45483430 Ki = 2 nM T27812 CG2SM9 45483458 Ki = 81 nM T27812 CFM9P8 45483465 Ki = 98 nM T27812 C5DS3M 45483506 Ki = 781 nM T27812 CHCA47 45483511 Ki = 53 nM T27812 CD5H2X 45483622 IC50 > 10000 nM T27812 C1Q8EH 45486492 IC50 = 2833 nM T27812 C0HSJ7 45486515 IC50 = 918 nM T27812 C0IZ7C 45486517 IC50 = 74 nM T27812 C7E0XV 45486600 IC50 = 298 nM T27812 CVW53R 45486602 IC50 = 50 nM T27812 C3HB5W 45486603 IC50 = 161 nM T27812 C0UV4I 45486616 IC50 = 2200 nM T27812 CR2J3T 45486621 IC50 = 251 nM T27812 CD8TC7 45486628 IC50 = 299 nM T27812 CMN6J2 45486630 IC50 = 95 nM T27812 COY84K 45486646 IC50 = 10 nM T27812 C8N6SO 45486651 IC50 = 31 nM T27812 CA60OT 45486819 Ki = 62 nM T27812 CQMJ83 45486820 Ki = 8 nM T27812 CJN7X0 45486824 Ki = 1 nM T27812 CSIO35 45486825 Ki = 10 nM T27812 CFCD10 45486840 Ki = 21 nM T27812 C49EAG 45486845 Ki = 41 nM T27812 C6ROX8 45486859 Ki = 1140 nM T27812 C6Q4AJ 45486879 Ki = 25 nM T27812 CY9ZD8 45486887 Ki = 5200 nM T27812 C9BSL5 45486891 Ki = 4 nM T27812 CB0JM3 45486892 Ki = 62 nM T27812 CO9JN6 45486893 Ki = 3 nM T27812 CI8NA1 45486898 Ki = 1200 nM T27812 C4H7OT 45486902 Ki = 0.4 nM T27812 CI89OX 45487689 IC50 = 10 nM T27812 CC75GW 45487699 IC50 = 12 nM T27812 CVM34I 45487708 IC50 > 400 nM T27812 CAIV28 45487720 IC50 = 58 nM T27812 CNFI42 45487726 IC50 = 10 nM T27812 CAO36Q 45487761 IC50 = 15 nM T27812 C80FMT 45487762 IC50 = 17 nM T27812 CL9SM3 45487783 IC50 = 9 nM T27812 CL1H2W 46200976 Ki = 7 nM T27812 C79ZBC 46200977 Ki = 12 nM T27812 CIV92F 46214153 Ki = 1 nM T27812 CI39BE 46216792 IC50 = 1.1 nM T27812 C62BEZ 46224739 Ki = 139 nM T27812 C5LTG9 46225164 Ki = 671 nM T27812 CQT3G4 46225165 Ki = 9 nM T27812 C5OC1A 46225166 Ki = 8 nM T27812 C1AM8J 46225207 Ki = 5 nM T27812 CNQ10M 46225208 Ki = 63 nM T27812 C5RH4O 46225261 Ki = 617 nM T27812 COI1K0 46225262 Ki = 1242 nM T27812 C8Z0DR 46225263 Ki = 31 nM T27812 CYE41P 46225264 Ki = 13 nM T27812 C2H1PN 46225309 Ki = 12 nM T27812 CUR54A 46225310 Ki = 20 nM T27812 CGY19F 46226540 Ki = 0.58 nM T27812 C79GDE 46226541 Ki = 4000 nM T27812 C0H7ID 46226542 Ki = 2500 nM T27812 C5TSH8 46226543 Ki = 3200 nM T27812 CL07MO 46226544 Ki = 1500 nM T27812 CMK1Z6 46226545 Ki = 2600 nM T27812 C1KSD4 46226546 Ki = 65 nM T27812 CED57N 46226547 Ki = 2100 nM T27812 C27DWI 46226548 Ki = 470 nM T27812 C3I4ZU 46226549 Ki = 250 nM T27812 C6UDJ2 46226550 Ki = 810 nM T27812 C8Q0JS 46226551 Ki = 270 nM T27812 C6SGC5 46226552 Ki = 730 nM T27812 C70RNJ 46226553 Ki = 340 nM T27812 C72NRZ 46226554 Ki = 160 nM T27812 C8FM7G 46226555 Ki = 62 nM T27812 CJS97C 46226556 Ki = 860 nM T27812 CB8XA5 46226557 Ki = 27 nM T27812 COC3L5 46226572 Ki = 0.86 nM T27812 CJKZ16 46226573 Ki = 3.5 nM T27812 CF6I8D 46226574 Ki = 20 nM T27812 CE0W4J 46227268 Ki = 127 nM T27812 CY5FD9 46227269 IC50 = 404 nM T27812 CY82LR 46227396 IC50 > 10000 nM T27812 C06QIT 46227754 Ki = 10 nM T27812 C30ZIR 46227757 Ki = 17 nM T27812 C4YLZ1 46227762 Ki = 61 nM T27812 C08ZOG 46227770 Ki = 30 nM T27812 CJ9OF6 46228636 Ki = 0.3162 nM T27812 CSNI09 46228719 Ki = 15.85 nM T27812 CG68MR 46228720 Ki = 1 nM T27812 C5NB2Z 46228786 Ki = 0.3162 nM T27812 C5JPE2 46229669 Ki = 13 nM T27812 C4B0FX 46229670 Ki = 7 nM T27812 C39VDA 46229671 Ki = 519 nM T27812 CS0EJ4 46229672 Ki = 401 nM T27812 C32VBR 46229686 Ki = 445 nM T27812 CN4HT2 46230756 Ki = 251 nM T27812 CHZA09 46230766 IC50 = 2.5 nM T27812 CW8P4O 46230826 IC50 = 3.9 nM T27812 CDU9Q3 46230827 IC50 = 4 nM T27812 C2GU4H 46230828 IC50 = 80 nM T27812 CG9WO4 46230829 IC50 = 7 nM T27812 C51XBZ 46230830 IC50 = 46 nM T27812 CTU39D 46230883 IC50 = 17 nM T27812 C51MFX 46230884 IC50 = 2.1 nM T27812 CZ8VP0 46230885 IC50 = 18 nM T27812 C0B5FP 46230886 IC50 = 7.6 nM T27812 CN2Z0F 46230887 IC50 = 76 nM T27812 CDL76I 46230888 IC50 = 17 nM T27812 C83HGU 46230935 IC50 = 8.1 nM T27812 CDN7E1 46230936 IC50 = 5.7 nM T27812 CSZ7B2 46230937 IC50 = 120 nM T27812 CI8O5W 46233622 IC50 = 329 nM T27812 C7OB2G 46235733 IC50 = 501.19 nM T27812 C42SVX 46700866 IC50 > 10000 nM T27812 CD0K6E 46700867 IC50 = 6700 nM T27812 CJ2D3O 46701015 IC50 = 48.98 nM T27812 CM04ZI 46701016 IC50 = 83.18 nM T27812 C0JWP5 46701017 IC50 = 3.631 nM T27812 C5H0MJ 46701086 IC50 = 114.82 nM T27812 C9HWI7 46701087 IC50 = 91.2 nM T27812 CVE5O1 46701088 IC50 = 107.15 nM T27812 C1VPM0 46701089 IC50 = 9.772 nM T27812 CQ8B6R 46701090 IC50 = 69.18 nM T27812 C6C0FS 46701091 IC50 = 45.71 nM T27812 CQ7S3X 46837648 IC50 = 4600 nM T27812 CL7VN1 46837649 IC50 = 390 nM T27812 CU7OG4 46837651 IC50 > 100000 nM T27812 C5WNL1 46837652 IC50 > 100000 nM T27812 COX2H5 46837653 IC50 > 100000 nM T27812 CWZY17 46837780 IC50 = 4600 nM T27812 CV2NT3 46837781 IC50 > 100000 nM T27812 CT83MU 46837782 IC50 > 100000 nM T27812 C5TY3Q 46837783 IC50 > 100000 nM T27812 CWJF83 46837784 IC50 > 100000 nM T27812 C0ZSY5 46837785 IC50 > 100000 nM T27812 CBQJ74 46837922 IC50 = 1800 nM T27812 C8UWQ2 46837923 IC50 = 300 nM T27812 CCX8T0 46837924 IC50 = 540 nM T27812 CBH49N 46837925 IC50 = 6480 nM T27812 CH76RQ 46855361 Ki = 79.43 nM T27812 CFJ3Q4 46855363 Ki = 50.12 nM T27812 CEG23T 46855638 Ki = 0.3981 nM T27812 CFW0B9 46855640 Ki = 15.85 nM T27812 CKS74N 46855641 Ki = 100 nM T27812 C7FPT6 46855642 Ki = 1 nM T27812 CZS2G8 46855643 Ki = 5.012 nM T27812 C9AG3X 46855785 Ki = 3.981 nM T27812 C2WKY8 46855786 Ki = 100 nM T27812 CB51DQ 46855787 Ki = 251.19 nM T27812 CHT1G5 46855789 Ki = 630.96 nM T27812 CLX6M3 46855790 Ki = 1.585 nM T27812 C0CG4F 46866510 Ki = 0.3162 nM T27812 C1OE2K 46877858 IC50 = 4087 nM T27812 C7PDE6 46877860 IC50 = 5500 nM T27812 C89FYG 46877878 IC50 = 1590 nM T27812 CT3R2F 46877879 IC50 = 1220 nM T27812 CHIW05 46880277 IC50 = 57 nM T27812 CK8A1O 46880462 Ki > 10000 nM T27812 C9KDP4 46880463 Ki > 10000 nM T27812 CODR73 46880498 Ki > 10000 nM T27812 CHJ5Y6 46880566 Ki > 10000 nM T27812 CE9PG2 46880567 Ki > 10000 nM T27812 C01PGO 46880568 Ki > 10000 nM T27812 CS7L4X 46880569 Ki > 10000 nM T27812 C0PXY7 46880628 Ki > 10000 nM T27812 CD37LU 46880629 Ki > 10000 nM T27812 CUY89F 46880630 Ki > 10000 nM T27812 C4P6XS 46880631 Ki > 10000 nM T27812 CJ53KF 46880672 Ki > 10000 nM T27812 CYJC08 46880673 Ki > 10000 nM T27812 C1RI9O 46880674 Ki > 10000 nM T27812 CMS27C 46882857 Ki = 6 nM T27812 CM45ZP 46882858 Ki = 3 nM T27812 C3IGF1 46882859 Ki = 54 nM T27812 CHLZ97 46882860 Ki = 6 nM T27812 C4B8EX 46882909 Ki = 11 nM T27812 CFY95C 46882910 Ki = 3 nM T27812 C6GJ1F 46882911 Ki = 15 nM T27812 C0SQX2 46882912 Ki = 10 nM T27812 CJ82WI 46882913 Ki = 25 nM T27812 CV94JW 46882937 Ki = 7 nM T27812 CM5Z4G 46882938 Ki = 1320 nM T27812 CJV6R1 46882939 Ki = 13 nM T27812 C60YMF 46883462 Ki = 29 nM T27812 C7J6GU 46883497 Ki = 16 nM T27812 C3F5AS 46883498 Ki = 15 nM T27812 CRSE34 46883499 Ki = 4 nM T27812 C0CX3O 46883500 Ki = 20 nM T27812 CZR76I 46888925 Ki = 538 nM T27812 C4Q3SD 46888926 Ki = 93 nM T27812 CH9S8A 46888927 Ki = 94 nM T27812 C8T6WQ 46888928 Ki = 1.9 nM T27812 CJY47V 46888983 Ki = 19 nM T27812 CJ6IB7 46888984 Ki = 20 nM T27812 C18KHC 46888985 Ki = 20 nM T27812 CK40FT 46888986 Ki = 22 nM T27812 CTJ1P2 46889013 Ki = 30 nM T27812 COPQ75 46889014 Ki = 0.26 nM T27812 CAM45V 46889015 Ki = 1.5 nM T27812 CZ3FI5 46889016 Ki = 1.7 nM T27812 C4B6ZE 46889041 Ki = 5 nM T27812 CH56AN 46890391 Ki = 18 nM T27812 CPDX34 46890392 Ki = 19 nM T27812 C0YGP2 46890393 Ki = 19 nM T27812 C61INJ 46890394 Ki = 8 nM T27812 CI14SE 46890441 Ki = 2 nM T27812 CP4GD3 46890442 Ki = 9 nM T27812 CQI2Y8 46890443 Ki = 19 nM T27812 CZ2MG7 46890444 Ki = 10 nM T27812 CP6A8K 46890445 Ki = 8 nM T27812 CD5J8B 46890446 Ki = 8 nM T27812 CYK9D2 46890489 Ki = 17 nM T27812 CCR04L 46890490 Ki = 12 nM T27812 CT4O9M 46890491 Ki = 9 nM T27812 CGPM19 46890493 Ki = 16 nM T27812 CJ6K2R 46891598 Ki = 16 nM T27812 C1JSH9 46899637 Ki = 5.012 nM T27812 C3MSL0 46899638 Ki = 6.31 nM T27812 CV3LP2 46899639 Ki = 12.59 nM T27812 CGHZ15 46899640 Ki = 10 nM T27812 CN9FC3 46900150 Ki = 19.95 nM T27812 C40ZJO 46900451 Ki = 19.95 nM T27812 CNC02A 46900453 Ki = 15.85 nM T27812 CTCH14 46900455 Ki = 31.62 nM T27812 CP41AQ 46900457 Ki = 12.59 nM T27812 CR3L4I 46900459 Ki = 199.53 nM T27812 CK17PA 46900606 Ki = 10 nM T27812 CQ2K1C 46900608 Ki = 50.12 nM T27812 C5ZT1B 46900610 Ki = 15.85 nM T27812 C1NAX4 46900612 Ki = 31.62 nM T27812 CT0SQ2 46900614 Ki = 39.81 nM T27812 CXD9S3 46900776 Ki = 15.85 nM T27812 C8I7SJ 46900778 Ki = 125.89 nM T27812 C7QDM9 46900782 Ki = 7.943 nM T27812 C15FMY 46900954 Ki = 15.85 nM T27812 C8W1FU 46900956 Ki = 19.95 nM T27812 CH35BV 46900958 Ki = 10 nM T27812 CJH50B 46905305 IC50 > 1000 nM T27812 CAT25E 46905306 IC50 > 1000 nM T27812 C2TP6B 46905307 IC50 = 20 nM T27812 CPN09J 46905308 IC50 > 1000 nM T27812 C4XF8B 46907064 IC50 = 2500 nM T27812 C9P5JV 46907065 IC50 = 15700 nM T27812 CC5VA8 46907097 IC50 = 2200 nM T27812 CRV5K0 46913908 Ki = 390 nM T27812 CZ2G1P 46914046 IC50 = 3400 nM T27812 C2ULG1 46927928 IC50 = 7096 nM T27812 CK21VU 46927929 IC50 = 54 nM T27812 C68AJP 46933238 Ki = 0.5012 nM T27812 CX7R3H 46933845 Ki > 10000 nM T27812 CAY75I 46934585 Ki = 1 nM T27812 C6J4TV 46946859 Ki = 16.5 nM T27812 CW8YC3 49765184 Ki = 7 nM T27812 C2LZJ0 49783209 Ki = 9006 nM T27812 C57SMG 49783415 Ki > 10000 nM T27812 C0TG6I 49783419 Ki > 10000 nM T27812 CO6W0D 49798171 Ki = 15.85 nM T27812 CHQ7I8 49798172 Ki = 79.43 nM T27812 CMBX16 49798173 Ki = 100 nM T27812 CMO8V7 49798193 Ki = 50.12 nM T27812 C60YCR 49798194 Ki = 3.162 nM T27812 C85KNS 49798241 Ki = 39.81 nM T27812 CQ4G1V 49798242 Ki = 158.49 nM T27812 C01JNE 49798243 Ki = 3.981 nM T27812 CC6MF8 49798244 Ki = 79.43 nM T27812 CYAS45 49798266 Ki = 1 nM T27812 C2UO0F 49799236 IC50 > 100000 nM T27812 C6FH8G 49799237 IC50 > 100000 nM T27812 CZ3US5 49799443 Ki = 100 nM T27812 CQH0U4 49799522 Ki = 31.62 nM T27812 CZ76MQ 49799633 IC50 = 360 nM T27812 CU28RO 49799634 IC50 > 100000 nM T27812 CN89XG 49799642 IC50 = 1565 nM T27812 C85MBT 49799643 IC50 = 334 nM T27812 CK6IA0 49799933 IC50 = 2200 nM T27812 C58AWR 49818125 Ki = 1.259 nM T27812 CDV79P 49818201 Ki = 2.089 nM T27812 CFX2Q0 49818202 Ki = 31.62 nM T27812 C23PXY 49818203 Ki = 10 nM T27812 CB6OA3 49836197 Ki > 70 nM T27812 CP87FO 49836198 Ki > 70 nM T27812 CU2NF0 49836199 Ki > 70 nM T27812 CFB53A 49836200 Ki > 70 nM T27812 CR40BA 49836386 IC50 = 0.22 nM T27812 CNSA40 49836387 IC50 = 0.97 nM T27812 CWO42Q 49836388 IC50 = 0.38 nM T27812 C5LF8M 49836389 IC50 = 1.3 nM T27812 CLY74X 49836390 IC50 = 2.4 nM T27812 CO7QU1 49836495 IC50 = 5.9 nM T27812 C0M5XC 49836496 IC50 = 0.63 nM T27812 CAFZ28 49836497 IC50 = 2.8 nM T27812 CZJV13 49852019 IC50 > 100000 nM T27812 CSL8M9 49852020 IC50 = 6.2 nM T27812 CWCY74 49852021 IC50 = 115 nM T27812 CI08OL 49852022 IC50 = 700 nM T27812 C1BH4A 49852023 IC50 = 105 nM T27812 C0VT3Z 49856376 Ki = 184 nM T27812 CV21GT 49856377 Ki = 631 nM T27812 CIA24C 49863566 IC50 = 860 nM T27812 CZB85K 49863567 IC50 = 375 nM T27812 C7V6WO 49863654 IC50 = 23 nM T27812 CH36GC 49863692 IC50 = 225 nM T27812 C39VLG 49863693 IC50 = 1259 nM T27812 CKF87D 49863694 IC50 = 183 nM T27812 CZF5Q2 49863695 IC50 = 22 nM T27812 CFTZ59 49863717 IC50 = 300 nM T27812 COR7M1 49863727 Ki = 357.4 nM T27812 C7CJ5W 49863728 Ki = 11.3 nM T27812 C9YS5V 49863729 Ki = 8.5 nM T27812 C7IK0Y 49863741 IC50 = 284 nM T27812 C1GR9V 49863742 IC50 = 225 nM T27812 CRQ7U4 49863743 IC50 = 1084 nM T27812 CO3K6A 49863748 Ki = 2.2 nM T27812 CK92TE 49863749 Ki = 147 nM T27812 CF2TO6 49863774 IC50 = 322 nM T27812 C7Y8OQ 49863775 IC50 = 1981 nM T27812 C24EAI 49863776 IC50 = 854 nM T27812 CM72WN 49863778 IC50 = 381 nM T27812 CZR6T8 49863794 IC50 = 82 nM T27812 CB13XF 49863795 IC50 = 163 nM T27812 C6GB5R 49863847 IC50 = 162 nM T27812 C8PQB0 49863849 IC50 = 78 nM T27812 C1EKY3 49863851 IC50 = 78 nM T27812 CS80EL 49863853 IC50 = 36 nM T27812 C4HB5K 49863957 IC50 = 78 nM T27812 C18ICN 49863958 IC50 = 908 nM T27812 C8H6GV 49863959 IC50 = 252 nM T27812 CMRQ30 49863961 IC50 = 45 nM T27812 CFZ39O 49865822 Ki = 0.5012 nM T27812 CT34HY 49865823 Ki = 7.943 nM T27812 CK7O1S 49865875 Ki = 1.995 nM T27812 CCH8T4 49865876 Ki = 0.3981 nM T27812 C8V3NG 49865877 Ki = 1.259 nM T27812 CEK89Q 49865878 Ki = 15.85 nM T27812 CZA5X4 49865879 Ki = 2.512 nM T27812 CD4LO5 49865880 Ki = 5.012 nM T27812 CZ2W8K 49865881 Ki = 794.33 nM T27812 C0R8AN 49865934 Ki = 1258.93 nM T27812 C9TN8D 49865935 Ki = 12.59 nM T27812 C3YJ4G 49865936 Ki = 1.995 nM T27812 CB5WR8 49865937 Ki = 6.31 nM T27812 C8LJ4H 49865983 Ki = 1 nM T27812 C1MPT6 49865984 Ki = 6.31 nM T27812 C62NWE 49865985 Ki = 1.995 nM T27812 C5H4AY 49865986 Ki = 0.1995 nM T27812 C90XRC 49865987 Ki = 5.012 nM T27812 CKMX26 49866033 IC50 = 279 nM T27812 CEFJ14 49866038 Ki = 12.59 nM T27812 CZ9I3O 49866039 Ki = 1 nM T27812 C96XFK 49866040 Ki = 31.62 nM T27812 C26NLJ 49866041 Ki = 0.631 nM T27812 CQHM34 49866042 Ki = 0.3981 nM T27812 CK1Y3B 49866085 IC50 = 660 nM T27812 C8JY3K 49866095 Ki = 1 nM T27812 C9N5CZ 49866096 Ki = 3.162 nM T27812 CC1L4U 49866097 Ki = 1.585 nM T27812 CV49QI 49866161 Ki = 0.3981 nM T27812 CF59UG 49866162 Ki = 3.162 nM T27812 C5N8KG 49866163 Ki = 0.631 nM T27812 C4F8UX 49866191 Ki = 3.981 nM T27812 C2RY0J 50878551 Ki = 501.19 nM T27812 C1W6TV 50898777 Ki > 10000 nM T27812 CXMZ73 50898778 Ki > 10000 nM T27812 CYGD56 50899654 IC50 = 289 nM T27812 CBLK68 50899745 IC50 = 644 nM T27812 CJI9U2 50899747 IC50 = 881 nM T27812 CU7TK4 50899749 IC50 = 1014 nM T27812 C67IRJ 50908804 Ki = 0.2512 nM T27812 CLOB24 50908805 Ki = 1.259 nM T27812 CA89QH 50914389 Ki = 8.44 nM T27812 C2CYL1 50917604 Ki = 3211 nM T27812 C0C9HA 50917605 Ki = 7.4 nM T27812 C9U6BI 50917780 Ki = 15315 nM T27812 C6JNK5 50917781 Ki = 10.5 nM T27812 C1C9JT 50917784 Ki = 29104 nM T27812 C1BMO5 50917785 Ki = 20.6 nM T27812 C8J5MB 50941458 IC50 = 3 nM T27812 CJP82R 50941459 IC50 = 650 nM T27812 CJ43IF 50941460 IC50 = 20 nM T27812 CIGJ83 50942207 IC50 > 1000 nM T27812 CK4HM2 50942208 IC50 > 1000 nM T27812 C2SHO8 50993865 IC50 = 107 nM T27812 CX48AD 51002362 Ki > 10000 nM T27812 C6LVM3 51003382 Ki = 1160 nM T27812 CIW56N 51003383 Ki > 4900 nM T27812 CQ8KP7 51003749 IC50 = 2100 nM T27812 CE4KP1 51050257 Ki > 10000 nM T27812 CYR7P8 51346818 IC50 = 169 nM T27812 CD4B6S 51346820 IC50 = 34 nM T27812 CUQ53T 52918018 IC50 = 4500 nM T27812 CTP6U5 52918019 IC50 = 4400 nM T27812 CX5ZB8 52940714 IC50 = 2096 nM T27812 C9C0NB 52940734 Ki = 47 nM T27812 C0UXM7 52941358 Ki = 48.1 nM T27812 CTM81E 52941423 Ki = 292 nM T27812 C8E1MB 52941809 Ki = 24 nM T27812 CE26GV 52941856 IC50 = 730 nM T27812 CH86KJ 52941866 IC50 = 347 nM T27812 CX9AF4 52942551 Ki = 251.19 nM T27812 CE6R7D 52942615 Ki = 194 nM T27812 CR0G5U 52942644 Ki = 199.53 nM T27812 CGC90M 52943149 Ki = 2.4 nM T27812 CCF97B 52943811 Ki = 100 nM T27812 C2FG9O 52943861 Ki = 12.59 nM T27812 C9G4CI 52943891 Ki = 3.981 nM T27812 CZ21PJ 52944292 IC50 = 646 nM T27812 CBU2Z6 52944379 Ki = 1040 nM T27812 CCVP06 52944840 Ki = 2.512 nM T27812 C59ASG 52945060 Ki = 437 nM T27812 CL0BQ2 52945369 IC50 = 600 nM T27812 C2TK7W 52945494 IC50 = 1213 nM T27812 CPD0Y9 52945500 IC50 = 394 nM T27812 CL7OG0 52945537 IC50 = 537 nM T27812 CHFI03 52945539 IC50 = 6374 nM T27812 C4SH8M 52945840 Ki = 8.81 nM T27812 CJ49MX 52946290 Ki = 15.85 nM T27812 CJV4D0 52946564 IC50 = 240 nM T27812 CRIV53 52946792 Ki = 21.4 nM T27812 C4S8JC 52946835 Ki = 504 nM T27812 CS3OD1 52947342 Ki = 230 nM T27812 CCOQ59 52947343 Ki = 213 nM T27812 C6YB2T 52947380 Ki = 67.7 nM T27812 CK5ER0 52947414 Ki = 12.59 nM T27812 CAVB03 52947615 Ki = 0.5012 nM T27812 C1HRK4 52947622 Ki = 0.5012 nM T27812 CQCB97 52947785 IC50 = 340 nM T27812 C0K8CF 52947796 IC50 = 8000 nM T27812 CRH1P6 52947969 IC50 = 588 nM T27812 CD17LV 52948101 Ki = 174 nM T27812 C7IR4Q 52948256 Ki = 13.6 nM T27812 CJ6OP5 52948620 Ki = 45.6 nM T27812 C4ZC1K 52948697 Ki = 12.59 nM T27812 C8XB1M 52949040 IC50 = 2500 nM T27812 CFN80U 52949206 IC50 = 892 nM T27812 CLOB90 52949351 Ki = 118 nM T27812 C0RUM1 52949810 Ki = 96.3 nM T27812 CS6O4B 52949885 Ki = 388 nM T27812 CILY85 52950060 Ki = 104 nM T27812 CPVM58 52950169 Ki = 20.2 nM T27812 C42NYA 53248999 Ki = 63.1 nM T27812 CKS81C 53316705 IC50 > 10000 nM T27812 CVZ7U8 53316706 IC50 > 7000 nM T27812 CB01DE 53316707 IC50 > 4000 nM T27812 C6IHN7 53316708 IC50 > 10000 nM T27812 CKG01N 53316721 Ki = 0.08 nM T27812 CGQJ07 53316788 Ki = 3250 nM T27812 CR41UN 53316822 IC50 = 7 nM T27812 CL78NK 53316823 IC50 = 54 nM T27812 CB86XC 53316913 IC50 = 881 nM T27812 CE26AQ 53317143 IC50 = 156 nM T27812 C2V6WS 53317144 IC50 = 299 nM T27812 C9L6YK 53317145 IC50 = 278 nM T27812 CST69D 53317146 IC50 = 55 nM T27812 CS9Z0R 53317167 IC50 = 767 nM T27812 CH76LD 53317168 IC50 = 31 nM T27812 C63XCS 53317410 IC50 = 105 nM T27812 C9RNL2 53317411 IC50 = 48 nM T27812 CPK1R2 53317591 IC50 > 10000 nM T27812 CU2R4V 53317717 IC50 > 10000 nM T27812 CZTW58 53317736 Ki > 4710 nM T27812 CIK7D3 53317746 IC50 > 10000 nM T27812 CW0G5B 53318001 IC50 > 10000 nM T27812 C7APQ5 53318002 IC50 > 10000 nM T27812 CRHA45 53318003 IC50 > 10000 nM T27812 C1HO3W 53318004 IC50 > 10000 nM T27812 C68GHK 53318005 IC50 > 10000 nM T27812 CW70NZ 53318092 Ki > 4650 nM T27812 C7PC1G 53318093 Ki > 4710 nM T27812 CQ37BK 53318094 Ki = 2230 nM T27812 C8RLQ9 53318095 Ki > 4530 nM T27812 C85UKZ 53318218 IC50 = 5655 nM T27812 CFHE24 53318434 IC50 = 2240 nM T27812 CI49RQ 53318452 IC50 = 2723 nM T27812 CWHC74 53318453 IC50 = 1530 nM T27812 CD0Y4B 53318705 IC50 = 4624 nM T27812 CE1W5G 53318706 IC50 = 2610 nM T27812 C8C7YZ 53318707 IC50 > 10000 nM T27812 C8PAY5 53318980 IC50 = 1079 nM T27812 CZ0M8J 53319021 IC50 = 42 nM T27812 C8V1AW 53319232 IC50 = 2400 nM T27812 C7BY4O 53319345 IC50 > 10000 nM T27812 C5FRP2 53319428 Ki > 4710 nM T27812 CY65NV 53319429 Ki > 4620 nM T27812 C1MD0J 53319430 Ki = 94 nM T27812 C1E7BF 53319431 Ki > 4710 nM T27812 C2OJW5 53319432 Ki > 4530 nM T27812 CT0W3X 53319433 Ki > 6130 nM T27812 C8EKT2 53319478 IC50 = 3 nM T27812 C79JCL 53319479 IC50 = 2 nM T27812 CK2G3D 53319480 IC50 = 23 nM T27812 CVXT03 53319481 IC50 = 16 nM T27812 C90TZS 53319482 IC50 = 2495 nM T27812 CJH1M0 53319767 IC50 = 8571 nM T27812 CZ6L5C 53319784 IC50 = 305 nM T27812 CE6V4A 53319785 IC50 = 286 nM T27812 C63JGV 53319832 IC50 = 6 nM T27812 CVF5U0 53319835 IC50 = 96 nM T27812 CXF1S4 53320328 IC50 = 9 nM T27812 CODA90 53320569 Ki > 10000 nM T27812 CZE80U 53320651 IC50 > 10000 nM T27812 CQC23J 53320652 IC50 = 755 nM T27812 C19ZWJ 53320686 IC50 = 2550 nM T27812 CB84NG 53320778 IC50 = 125 nM T27812 C8JX4C 53320779 IC50 = 1 nM T27812 CP7RZ3 53320780 IC50 = 61 nM T27812 CL67KH 53320781 IC50 = 970 nM T27812 CK5C0S 53320864 IC50 = 135 nM T27812 CQ90IR 53321058 IC50 = 19 nM T27812 CZ7NM6 53321059 IC50 = 1870 nM T27812 CXY92R 53321081 IC50 = 57 nM T27812 CS42VL 53321082 IC50 = 224 nM T27812 CO7L6Z 53321083 IC50 = 3 nM T27812 CSY1K4 53321125 IC50 = 5900 nM T27812 CAJ4L7 53321331 IC50 = 208 nM T27812 CMZ7F8 53321332 IC50 = 2550 nM T27812 CZEF75 53321509 IC50 > 10000 nM T27812 C1AI0C 53321510 IC50 > 10000 nM T27812 C34ORB 53321945 IC50 > 10000 nM T27812 C6ND9H 53321946 IC50 > 10000 nM T27812 C4X3IS 53321979 IC50 = 116 nM T27812 CLQ85U 53322027 Ki = 2040 nM T27812 C53HJK 53322028 Ki > 4690 nM T27812 CLD82J 53322084 IC50 = 6 nM T27812 C7QF2E 53322085 IC50 = 20 nM T27812 CY09UA 53322086 IC50 = 1956 nM T27812 CBUT35 53322087 IC50 = 2827 nM T27812 CXL8W9 53322200 IC50 = 624 nM T27812 CE63PO 53322201 IC50 = 369 nM T27812 C3M9SC 53322397 IC50 = 158 nM T27812 CLT3Q2 53322398 IC50 = 651 nM T27812 CZLT60 53322409 IC50 = 145 nM T27812 CLZ41J 53322410 IC50 = 249 nM T27812 C3YWZ5 53322451 IC50 = 12 nM T27812 CZ92BF 53322452 IC50 > 10000 nM T27812 C5G8RQ 53322642 IC50 = 8981 nM T27812 CV49EH 53322836 IC50 = 766 nM T27812 CRUF31 53322954 Ki > 4710 nM T27812 C3HKJ0 53323299 IC50 > 10000 nM T27812 C6ZFR5 53323300 IC50 > 2000 nM T27812 CK6U0Y 53323301 IC50 > 10000 nM T27812 CGA5R8 53323302 IC50 > 10000 nM T27812 CND26W 53323338 IC50 = 436 nM T27812 C6KAN9 53323339 IC50 = 5558 nM T27812 C2OB7G 53323389 Ki > 4620 nM T27812 C4UBX5 53323390 Ki > 4610 nM T27812 C1WU4E 53323391 Ki > 4710 nM T27812 CGN6Z3 53323531 IC50 = 7644 nM T27812 CAQ07J 53323532 IC50 = 136 nM T27812 C1GZ3B 53323533 IC50 = 25 nM T27812 C4D1LX 53323761 IC50 = 9674 nM T27812 CPKM07 53323762 IC50 = 7932 nM T27812 CQW2S7 53323771 IC50 < 1 nM T27812 CO7TC1 53323812 IC50 = 7100 nM T27812 CDRV76 53323814 IC50 = 150 nM T27812 C32YWL 53324045 Ki = 1180 nM T27812 C98OKX 53324333 IC50 = 33 nM T27812 C46XAC 53324366 IC50 = 985 nM T27812 CR4W9L 53324553 Ki > 10000 nM T27812 CCK4T2 53324628 IC50 > 10000 nM T27812 CW58QL 53324656 IC50 = 128 nM T27812 CFJ1B0 53324709 Ki > 6280 nM T27812 C5I1FG 53324762 IC50 = 108 nM T27812 C94GOI 53324763 IC50 = 19 nM T27812 COP3J6 53324764 IC50 = 311 nM T27812 CE7DZ0 53324844 IC50 = 43 nM T27812 CB34ZM 53325028 IC50 = 898 nM T27812 CY9H2U 53325042 IC50 = 689 nM T27812 CRQF15 53325242 Ki = 428 nM T27812 C3QNR2 53325463 IC50 = 132 nM T27812 CAGT23 53325525 IC50 > 10000 nM T27812 CZN8B4 53325581 IC50 = 8 nM T27812 COZ1W9 53325647 IC50 = 86 nM T27812 C1N7XO 53325966 IC50 = 7 nM T27812 CZ69OW 53326010 Ki = 2670 nM T27812 CZ1U9T 53326011 Ki = 1710 nM T27812 CM7YA0 53326118 IC50 = 106 nM T27812 CJ6G7X 53326119 IC50 = 1245 nM T27812 CTH12B 53326554 IC50 = 905 nM T27812 C0M5WU 53391513 IC50 = 147.91 nM T27812 C8DR9L 53391514 IC50 = 128.82 nM T27812 C7GH1I 53391515 IC50 = 34.67 nM T27812 C3BX4K 53391516 IC50 = 162.18 nM T27812 C5B1ST 53391517 IC50 = 6.918 nM T27812 CQYB97 53391614 IC50 = 1096.48 nM T27812 CK3D9F 53391615 IC50 = 4.467 nM T27812 C3S5QX 53391616 IC50 = 691.83 nM T27812 CI3T5Y 53391617 IC50 = 331.13 nM T27812 CKOD62 53391618 IC50 = 3.548 nM T27812 CD24UN 53391714 IC50 = 14.45 nM T27812 CA0GN6 53391715 IC50 = 33.11 nM T27812 CQ4E2W 53391716 IC50 = 12.59 nM T27812 C64TJO 53391717 IC50 = 13.49 nM T27812 C3Q6IL 53391718 IC50 = 120.23 nM T27812 C7UBN1 53392848 IC50 = 1819.7 nM T27812 CB5JU8 53392849 IC50 = 338.84 nM T27812 C0JI1M 53392850 IC50 = 5.495 nM T27812 CPIT32 53392851 IC50 = 660.69 nM T27812 C8K1TZ 53392852 IC50 = 48.98 nM T27812 CS7TE6 53392939 IC50 = 346.74 nM T27812 CT7U5L 53392940 IC50 = 1230.27 nM T27812 CMOZ61 53475319 Ki = 32 nM T27812 CDV82B 53492877 IC50 = 6410 nM T27812 C6Q3GO 54141274 Ki = 6.2 nM T27812 CPH4J9 54147697 Ki = 62 nM T27812 C43VJF 54296648 IC50 = 3790 nM T27812 CHE5Q4 54380151 Ki = 17 nM T27812 CNG7U0 54434812 Ki = 29830 nM T27812 C48CEL 54576149 IC50 = 21.6 nM T27812 C6PDR1 54576153 IC50 = 6 nM T27812 CX4OJ6 54576369 IC50 = 201 nM T27812 CA0O2M 54576371 IC50 = 70.3 nM T27812 CY67DI 54576594 IC50 = 7.59 nM T27812 CWUK35 54576597 IC50 = 16.6 nM T27812 C40IGO 54576800 IC50 = 6 nM T27812 CP4CV6 54576803 IC50 = 6.3 nM T27812 C4H3DT 54576804 IC50 = 150.1 nM T27812 CG24OE 54577010 IC50 = 5 nM T27812 CYZX34 54577012 IC50 = 16 nM T27812 C2WQE9 54577014 IC50 = 16.8 nM T27812 C83FGA 54577018 IC50 = 436.2 nM T27812 CWA58G 54577234 IC50 = 20.5 nM T27812 CA83GC 54577236 IC50 = 50.5 nM T27812 CJA0P6 54577243 IC50 = 12.6 nM T27812 C0NBJ7 54577435 IC50 = 9 nM T27812 CYW50O 54577439 IC50 = 28 nM T27812 C8YAZ5 54577443 IC50 = 31.1 nM T27812 C3P0LZ 54577446 IC50 = 9.3 nM T27812 CA94CQ 54577447 IC50 = 0.64 nM T27812 CE64WZ 54577448 IC50 = 5.08 nM T27812 CJS4H9 54577449 IC50 = 0.75 nM T27812 CMR6C3 54577665 IC50 = 13 nM T27812 CS9G8L 54577668 IC50 = 12 nM T27812 CA8J7E 54577670 IC50 = 10.3 nM T27812 C3P2KF 54577879 IC50 = 42.6 nM T27812 C9GFP0 54577882 IC50 = 6.9 nM T27812 C6KY9M 54577886 IC50 = 21.6 nM T27812 CES29I 54578098 IC50 = 6.6 nM T27812 CQ67LT 54578099 IC50 = 188 nM T27812 CAPC31 54578102 IC50 = 153.2 nM T27812 C12XBJ 54578547 IC50 = 10 nM T27812 CP24ZC 54579002 IC50 = 6.08 nM T27812 CXQK40 54579004 IC50 = 5 nM T27812 CZC81X 54579005 IC50 = 185 nM T27812 CSW18T 54579229 IC50 = 5 nM T27812 C5HC0P 54579233 IC50 = 19.1 nM T27812 CA4E9U 54579450 IC50 = 10.4 nM T27812 C3L1IB 54579451 IC50 = 1262 nM T27812 CEY2B8 54583277 IC50 = 1500 nM T27812 CF5Q0W 54583932 IC50 = 5700 nM T27812 C6ME0B 54584239 IC50 = 2900 nM T27812 CY4F0W 54584873 IC50 = 10000 nM T27812 CL5I1R 54753271 Ki = 295 nM T27812 C4URA5 54756923 IC50 = 5100 nM T27812 CYS19X 54756924 IC50 = 1775 nM T27812 CLC71N 54756925 IC50 = 1030 nM T27812 CT5F4Z 54757021 IC50 = 992 nM T27812 CPW0G4 54757022 IC50 = 8347 nM T27812 CYX2L8 54757023 IC50 = 806 nM T27812 CCZ97U 54757024 IC50 = 5790 nM T27812 COJ0T5 54757025 IC50 = 6770 nM T27812 C13SMB 54757119 IC50 = 749 nM T27812 C4S6UM 54757121 IC50 = 4128 nM T27812 CP5S0U 54757122 IC50 = 1400 nM T27812 CB87MF 54766009 IC50 = 501.4 nM T27812 C93WMS 54767239 IC50 = 399.3 nM T27812 CLV3N6 54767240 IC50 = 378.5 nM T27812 CZ47UJ 54767241 IC50 = 389.4 nM T27812 C5RX1P 54767242 IC50 = 546.1 nM T27812 C32NWX 54767413 IC50 = 425.3 nM T27812 C6ASW2 54767576 IC50 = 401 nM T27812 C45SEW 54767744 IC50 = 449.2 nM T27812 C3KV8R 54767747 IC50 = 1187.8 nM T27812 CO6CJ2 54767906 IC50 = 337.6 nM T27812 C9X4CE 56643874 EC50 = 714000 nM T27812 CMJ32F 56659126 Ki = 0.5012 nM T27812 CQ6XM7 56659146 Ki = 3.162 nM T27812 CFT9V8 56659147 Ki = 1.995 nM T27812 CO0GR7 56659199 Ki = 0.5012 nM T27812 CC26HR 56659200 Ki = 1.995 nM T27812 CGID30 56659201 Ki = 0.7943 nM T27812 CG0M7T 56662629 Ki = 0.2512 nM T27812 CP2ZS4 56662647 Ki = 1.259 nM T27812 C8NIZ3 56662648 Ki = 0.1995 nM T27812 CN7WB5 56662696 Ki = 0.2512 nM T27812 CD9F3J 56662697 Ki = 1 nM T27812 C5HF9D 56666091 Ki = 2.512 nM T27812 C9RE3V 56669493 Ki = 0.3981 nM T27812 CK3R7P 56669494 Ki = 3.981 nM T27812 CVRH79 56669561 Ki = 0.1 nM T27812 CC9XR7 56669562 Ki = 0.2512 nM T27812 CXE9A8 56669563 Ki = 0.1995 nM T27812 CNK39V 56673078 Ki = 6.31 nM T27812 C93KBW 56679646 Ki = 0.7943 nM T27812 CAR8M5 56679647 Ki = 2.512 nM T27812 CN1C3K 56679724 Ki = 7.943 nM T27812 CET3N2 56682964 Ki = 1.995 nM T27812 CK73UC 56683046 Ki = 0.3981 nM T27812 CZR91E 56683047 Ki = 7.943 nM T27812 C60IBF 56683048 Ki = 1.995 nM T27812 C90DOS 56942993 IC50 = 4.9 nM T27812 CB0P9N 56944383 IC50 > 1000 nM T27812 C1ST9U 56944860 Ki = 5.1 nM T27812 CQKL90 56944861 Ki = 5.2 nM T27812 CS5J6Y 56944862 Ki = 6.1 nM T27812 CFLB40 56944863 Ki = 2.8 nM T27812 C53OTR 56944864 Ki = 3.9 nM T27812 C5T3RI 56944951 Ki = 4.8 nM T27812 CR6H7U 56944952 Ki = 4.1 nM T27812 C1Y2RP 56944953 Ki = 4.6 nM T27812 C1BH7I 56944954 Ki = 3.5 nM T27812 CTK9I8 56944955 Ki = 2.7 nM T27812 CCF1A5 56944956 Ki = 3.6 nM T27812 C2YVT8 56945042 Ki = 6 nM T27812 CNI2G3 56945043 Ki = 3.3 nM T27812 CZI53T 56961001 IC50 = 200 nM T27812 C1TC7Q 56963799 Ki > 10000 nM T27812 CPT03G 57300602 Ki = 54 nM T27812 C4E1NK 57331209 IC50 = 9100 nM T27812 CATM39 57390694 Ki = 34 nM T27812 C6S0IE 57390695 Ki = 65 nM T27812 CCJ93V 57391031 Ki = 10298 nM T27812 C9LX1S 57391709 Ki > 1000 nM T27812 CMNZ07 57394992 IC50 = 100 nM T27812 C6SZ4E 57396296 Ki = 11 nM T27812 CJ41PW 57399432 Ki = 65 nM T27812 C92HON 57402951 Ki = 5.3 nM T27812 CX0B5M 57403525 Ki = 1867 nM T27812 C4N3VY 57403918 Ki = 251 nM T27812 CHU5T7 57523687 IC50 > 10 nM T27812 C3J9UN 57565074 IC50 = 51 nM T27812 CHB3D6 58405078 Ki = 27 nM T27812 CX2HU7 58405183 Ki = 124 nM T27812 CZI37P 58760107 Ki = 0.34 nM T27812 C0WJ4E 58954830 IC50 = 44 nM T27812 CSF52J 58954867 IC50 = 34 nM T27812 C9ZP3D 58954900 IC50 = 7 nM T27812 CHQE32 58954945 IC50 = 1187 nM T27812 CXH19J 59472574 IC50 = 32 nM T27812 CK6W7I 59536635 IC50 = 1.9 nM T27812 CA36QL 59800034 IC50 = 90300 nM T27812 CB9GC6 60165412 Ki = 298 nM T27812 CI5PM3 60165413 Ki = 64 nM T27812 C2Q5VD 60165416 Ki = 166 nM T27812 C31PEN 60165535 Ki = 1325 nM T27812 CP60YF 60165537 Ki = 186 nM T27812 CP1DR8 60165539 Ki = 491 nM T27812 C85OTH 60165541 Ki = 706 nM T27812 CJDC53 60165545 Ki = 237 nM T27812 C3K5JN 60165681 Ki = 81 nM T27812 C5RUP6 60167166 Ki = 1184 nM T27812 CRH49P 60167309 Ki = 922 nM T27812 CX0NY3 60167310 Ki > 10000 nM T27812 COHK72 60167451 Ki = 565 nM T27812 C30SVG 60167452 Ki = 281.84 nM T27812 CW36YC 66561968 Ki > 10000 nM T27812 CGF3J5 66572162 IC50 = 255 nM T27812 C95BOS 66572285 IC50 = 768 nM T27812 CZL90M 66572393 IC50 = 171 nM T27812 C2UZ3A 66572397 IC50 = 337 nM T27812 CCR2I5 66572399 IC50 = 425 nM T27812 CEB79F 66572506 IC50 = 357 nM T27812 C35VKU 66572510 IC50 = 367 nM T27812 CN30YT 66800947 Ki = 5.3 nM T27812 CZ3MR6 66800959 Ki = 8.5 nM T27812 C92CMO 66800965 Ki = 3.2 nM T27812 C3K8DC 66801052 Ki = 5.7 nM T27812 C41VYW 66801295 Ki = 1.1 nM T27812 CR2N0J 66801344 Ki = 3.8 nM T27812 C3RX4C 66801425 Ki = 2.3 nM T27812 C7JD0I 66801429 Ki = 32 nM T27812 CN8OU1 66801430 Ki = 40 nM T27812 COR1H8 66801528 Ki = 1.7 nM T27812 C1F3YV 66801537 Ki = 2.7 nM T27812 C75WXP 66801561 Ki = 4.3 nM T27812 CC8JV6 66801624 Ki = 12 nM T27812 C3EI2F 66801625 Ki = 16 nM T27812 C0XG6B 66801701 Ki = 18 nM T27812 C42EBQ 66801837 Ki = 25 nM T27812 CW3AI2 66803474 Ki = 5 nM T27812 CPKH06 66803497 Ki = 2.3 nM T27812 CNJE57 66803500 Ki = 4.2 nM T27812 CN6FZ1 66803595 Ki = 2.2 nM T27812 CL8R5V 66975152 IC50 = 54 nM T27812 C0OC8T 66975291 IC50 > 1000 nM T27812 CCN1W5 66975591 IC50 = 130 nM T27812 C23DPF 66975638 IC50 = 350 nM T27812 C3W0XI 66975648 IC50 = 780 nM T27812 C51JHP 66975671 IC50 = 36 nM T27812 CV19LA 66975764 IC50 = 27 nM T27812 C50HKX 66975948 IC50 = 200 nM T27812 C0L2QJ 66976018 IC50 = 330 nM T27812 CE9A4J 66976134 IC50 > 1000 nM T27812 CZE5S6 66976296 IC50 = 85 nM T27812 C78MWK 66976356 IC50 = 67 nM T27812 C5EM9P 66976389 IC50 > 1000 nM T27812 CP3M9I 66976532 IC50 = 150 nM T27812 CAL40U 66976565 IC50 = 79 nM T27812 CI29HX 66976607 IC50 = 12 nM T27812 C6I7SV 66976613 IC50 = 97 nM T27812 C8LD7M 66976718 IC50 = 200 nM T27812 C6ON5Y 66976777 IC50 > 1000 nM T27812 CI8SB4 67320583 IC50 > 10000 nM T27812 C7A8HK 67395483 Ki = 10 nM T27812 CB05ID 67972431 IC50 > 10000 nM T27812 C0MYB6 68653619 Ki = 250 nM T27812 CNY0W5 68673707 IC50 = 210 nM T27812 C76ROM 68673872 IC50 = 11 nM T27812 CD3U6K 68731121 Ki = 320 nM T27812 CSF80C 68993720 IC50 = 31 nM T27812 CVZ51D 68993987 IC50 = 110 nM T27812 CN0MY2 68994312 IC50 = 5.3 nM T27812 CKTA56 68994365 IC50 = 250 nM T27812 CE1WF3 68994389 IC50 = 28 nM T27812 CN08VY 68994725 IC50 = 4.4 nM T27812 C0ZY9I 68994988 IC50 = 4.5 nM T27812 CR3H9X 68995479 IC50 = 260 nM T27812 C1LWS9 68995587 IC50 = 18 nM T27812 CDLR80 68995667 IC50 = 170 nM T27812 CCIV97 68995742 IC50 = 4.9 nM T27812 C2MK1S 68995928 IC50 = 67 nM T27812 C56VJS 68996260 IC50 = 24 nM T27812 CQ4Y2V 68996331 IC50 = 29 nM T27812 CHI19N 68996402 IC50 = 6.4 nM T27812 C17BRZ 68997664 IC50 = 10 nM T27812 CDT9Z5 68998740 IC50 = 6.9 nM T27812 CP0AR5 68999429 IC50 = 8.4 nM T27812 CN14QD 69000395 IC50 = 4.4 nM T27812 C6IP8Q 69082816 Ki = 390 nM T27812 CNM1U4 69397184 Ki = 2310 nM T27812 CKM14W 69432471 Ki = 98 nM T27812 CYM94S 70676472 IC50 = 44 nM T27812 C7J0FD 70676474 IC50 = 6.8 nM T27812 CLTA38 70676476 IC50 = 8.3 nM T27812 CMN57J 70676478 IC50 = 35 nM T27812 C9QZ7C 70676480 IC50 = 142 nM T27812 C09HRL 70681048 IC50 = 248 nM T27812 CURI86 70681049 IC50 > 3000 nM T27812 CIX1V8 70681050 IC50 > 3000 nM T27812 C17ITX 70681051 IC50 = 35 nM T27812 C4ZK7S 70681052 IC50 = 30 nM T27812 CU32RF 70681053 IC50 = 566 nM T27812 C4AVG9 70681054 IC50 > 1000 nM T27812 CU48EX 70681055 IC50 = 10 nM T27812 C7W3JA 70681326 Ki = 0.5012 nM T27812 C67CHV 70681491 Ki > 10000000 nM T27812 CT65MH 70681573 Ki = 4361 nM T27812 CIE30Z 70683174 IC50 > 3000 nM T27812 C7X4VF 70683175 IC50 = 32 nM T27812 CP07IW 70683176 IC50 > 1000 nM T27812 C39QGY 70683608 Ki > 10000000 nM T27812 C0G2XO 70683685 Ki > 10000 nM T27812 C7HM6W 70685249 IC50 = 870 nM T27812 CQ8Y0N 70685250 IC50 > 3000 nM T27812 CC2L8W 70685251 IC50 > 3000 nM T27812 CFQ1I9 70685252 IC50 = 287 nM T27812 CDI70T 70685253 IC50 = 142 nM T27812 C60SBP 70685515 Ki = 25.12 nM T27812 CCOR65 70685727 Ki = 1459000 nM T27812 C3UBM6 70687401 IC50 > 3000 nM T27812 C05OPN 70687402 IC50 = 78 nM T27812 C1CH5A 70687667 Ki = 31.62 nM T27812 CTVW13 70689263 IC50 > 10000 nM T27812 C7RA0K 70689264 IC50 > 10000 nM T27812 CKMJ68 70689265 Ki = 1000 nM T27812 C4E3BZ 70689455 IC50 > 3000 nM T27812 C3OJY2 70689456 IC50 > 3000 nM T27812 CU84XH 70689457 IC50 = 395 nM T27812 C8NH5V 70689458 IC50 = 640 nM T27812 CB58JU 70691565 IC50 = 242 nM T27812 C3KS4O 70691566 IC50 > 3000 nM T27812 C5JPR4 70691567 IC50 > 2000 nM T27812 C7R0NO 70691568 IC50 > 3000 nM T27812 CS08ZT 70691569 IC50 = 128 nM T27812 CF63DA 70691570 IC50 = 77 nM T27812 CP8ZB4 70691571 IC50 > 1000 nM T27812 CVF95N 70691572 IC50 = 79 nM T27812 CMH98F 70691573 IC50 > 1000 nM T27812 C59NVG 70691872 Ki = 0.2512 nM T27812 C4A7QI 70692139 Ki > 10000 nM T27812 C74NGV 70693417 Ki = 4700 nM T27812 CB3NW6 70693452 Ki = 1500 nM T27812 CP38FE 70693453 Ki = 250 nM T27812 C7RF8K 70693651 IC50 > 3000 nM T27812 C6R4EB 70693652 IC50 > 3000 nM T27812 CP5I2J 70693653 IC50 > 3000 nM T27812 CYS1E6 70693654 IC50 > 3000 nM T27812 CR30AX 70693655 IC50 > 3000 nM T27812 C8IQC6 70695563 Ki = 356 nM T27812 C5DP3J 70695564 Ki = 140 nM T27812 CRXH46 70695767 IC50 = 710 nM T27812 CJ01ST 70695768 IC50 > 1000 nM T27812 C25SJC 70695769 IC50 > 3000 nM T27812 CRS3M8 70695770 IC50 = 556 nM T27812 CFM5Z8 70695771 IC50 > 1000 nM T27812 CN9RQ3 70695772 IC50 > 1000 nM T27812 C37USC 70697274 Ki = 63 nM T27812 CB9H4S 70697574 Ki = 376 nM T27812 CKD60A 70789640 Ki = 2495 nM T27812 CBDL19 70792359 IC50 = 898 nM T27812 CI93FE 70963695 IC50 = 5500 nM T27812 C2FN8M 71134973 IC50 = 35 nM T27812 CC43QK 71151588 Ki > 1000 nM T27812 C5BER9 71332336 IC50 = 1906 nM T27812 C6VL7X 71449080 Ki = 0.4 nM T27812 C9VZ8J 71450550 Ki = 548 nM T27812 C87FQH 71450609 Ki = 1470 nM T27812 C5IN6O 71450695 Ki = 58 nM T27812 CH3TV9 71450696 Ki = 2241 nM T27812 C97MYL 71450697 Ki = 52 nM T27812 C68BJU 71450818 IC50 = 64 nM T27812 CGQ0R2 71450907 Ki = 16 nM T27812 C6ZWV2 71452383 Ki = 4274 nM T27812 C01RKV 71452519 Ki = 827 nM T27812 C9WLY7 71452692 Ki = 9.24 nM T27812 CN4AJ2 71454274 Ki = 6.5 nM T27812 CE0R9D 71454275 Ki = 3512 nM T27812 C3S5EJ 71454276 Ki = 127 nM T27812 C0R2UV 71454458 Ki = 3.77 nM T27812 C6G2HC 71455894 Ki = 4421 nM T27812 CT2Z8R 71456033 Ki = 45 nM T27812 CD8O2C 71456208 Ki = 0.58 nM T27812 CUX98O 71456238 Ki = 104 nM T27812 COG3Y0 71456239 Ki = 106 nM T27812 CYR3D4 71456240 Ki = 7.3 nM T27812 C7MNB5 71457264 Ki = 1942 nM T27812 C6X1GN 71457767 Ki = 231 nM T27812 C8YD9T 71457837 Ki = 45 nM T27812 C3GKR6 71458006 Ki = 0.75 nM T27812 C87FDI 71458022 Ki = 590 nM T27812 COT5U4 71458045 IC50 = 18 nM T27812 CP16SV 71458086 IC50 = 290 nM T27812 C3OR6K 71459910 Ki = 7.18 nM T27812 CR3LH2 71461647 Ki = 1.4 nM T27812 CX69JF 71461719 IC50 = 7038 nM T27812 CD3L7R 71463125 Ki = 352 nM T27812 CUG7M5 71463194 Ki = 5638 nM T27812 C1XUO3 71463195 Ki = 122 nM T27812 C7IE9K 71463196 Ki = 23830 nM T27812 C6EF4I 71463197 Ki = 130 nM T27812 C4RAQ6 71518063 Ki = 225 nM T27812 CL8CK2 71521332 Ki = 0.03 nM T27812 CO26TC 71541094 Ki = 260 nM T27812 CE8YO0 71541095 Ki = 140 nM T27812 CN79ZY 71541096 Ki = 150 nM T27812 CNCR14 71541097 Ki = 540 nM T27812 CW34SU 71541098 Ki = 100 nM T27812 CKW24J 71541099 Ki = 83 nM T27812 C0ZL6O 71541186 Ki = 130 nM T27812 C92PZK 71541187 Ki = 270 nM T27812 C0T4RD 71541188 Ki = 800 nM T27812 CB91FO 71541189 Ki = 220 nM T27812 CY5E0J 71541190 Ki = 220 nM T27812 C4XK1S 71541191 Ki = 420 nM T27812 C32HNI 71541192 Ki = 63 nM T27812 C9C0JU 71541193 Ki = 600 nM T27812 CD1T5J 71541195 Ki = 1500 nM T27812 CQ81HF 71541289 Ki = 240 nM T27812 CU53JE 71541292 Ki = 230 nM T27812 CR7E4G 71541370 IC50 = 23 nM T27812 C9IE3U 71541371 IC50 = 3.1 nM T27812 CFO83N 71541372 IC50 = 6.3 nM T27812 CI6J5K 71541373 IC50 = 6.4 nM T27812 CC7YB2 71541376 IC50 = 2.2 nM T27812 CWT0Y3 71541468 IC50 = 12 nM T27812 CGJ86B 71541469 IC50 = 8.9 nM T27812 C0CBT4 71541470 IC50 = 10 nM T27812 CQ8JN9 71541471 IC50 = 12 nM T27812 CZV7N9 71541472 IC50 = 28 nM T27812 CL20CV 71541473 IC50 = 16 nM T27812 C6J9NY 71541572 IC50 = 5.6 nM T27812 CS0J6B 71541573 IC50 = 56 nM T27812 C5CO8Z 71541574 IC50 = 1.5 nM T27812 CI90PK 71541575 IC50 = 1.6 nM T27812 C4FS8Z 71541576 IC50 = 32 nM T27812 CSI37G 71541577 IC50 = 9.1 nM T27812 C5D6IE 71541687 IC50 = 8.3 nM T27812 C4A7KU 71550921 EC50 = 190 nM T27812 CLXR53 71560658 IC50 = 6000 nM T27812 C86MSF 71560659 IC50 = 4800 nM T27812 C7DPJ1 71560779 IC50 = 5500 nM T27812 C3XF2B 71560781 IC50 = 46000 nM T27812 C6B3CF 71562265 IC50 = 158.49 nM T27812 C9V0FZ 71562266 IC50 = 158.49 nM T27812 C49VSK 71562370 IC50 = 125.89 nM T27812 COFY97 71562371 IC50 = 63.1 nM T27812 C1JCZ5 71562372 IC50 = 12.59 nM T27812 CXR0E7 71562373 IC50 = 125.89 nM T27812 C4PDM8 71562374 IC50 = 3.981 nM T27812 C3L9HK 71562375 IC50 = 31.62 nM T27812 CX7VK3 71562376 IC50 = 2.512 nM T27812 CHW7K1 71562377 IC50 = 7.943 nM T27812 CK95GV 71562472 IC50 = 1.259 nM T27812 C4NS5W 71562473 IC50 = 19.95 nM T27812 C6X9SM 71562474 IC50 = 0.631 nM T27812 C1H4KQ 71562475 IC50 = 1.995 nM T27812 C6X3BP 71562476 IC50 = 63.1 nM T27812 CH49FE 71562477 IC50 = 10 nM T27812 CU1CZ6 71562478 IC50 = 0.7943 nM T27812 CPAY18 71562479 IC50 = 3.162 nM T27812 CY39RM 71562586 IC50 = 10 nM T27812 C4F2UW 71562587 IC50 = 39.81 nM T27812 CI3KA2 71562588 IC50 = 6.31 nM T27812 C13NIO 71562589 IC50 = 158.49 nM T27812 CKPH80 71562590 IC50 = 3.981 nM T27812 C0NIA6 71562591 IC50 = 15.85 nM T27812 CRCT65 71562592 IC50 = 1.259 nM T27812 C1XQ5M 71562593 IC50 = 0.631 nM T27812 CFQP86 71562712 IC50 = 1.585 nM T27812 CPDV40 71562713 IC50 = 1 nM T27812 CP2N3Y 71562714 IC50 = 25.12 nM T27812 CS59VG 71562715 IC50 = 1.585 nM T27812 CE7X9R 71562716 IC50 = 3.981 nM T27812 CP20LV 71562717 IC50 = 3.981 nM T27812 CQU78X 71562718 IC50 = 63.1 nM T27812 CCO48Y 71562719 IC50 = 3.981 nM T27812 CSYR25 71562833 IC50 = 15.85 nM T27812 CF0R4S 71562834 IC50 = 5.012 nM T27812 C5NO2C 71562835 IC50 = 6.31 nM T27812 C2UQD4 71562836 IC50 = 79.43 nM T27812 C1Q4JZ 71562837 IC50 = 5.012 nM T27812 CQ3L2J 71583092 IC50 = 970 nM T27812 CD0P5Z 71583093 IC50 > 1000 nM T27812 CER9H2 71583094 IC50 = 140 nM T27812 CK51UY 71583095 IC50 = 490 nM T27812 CJ8TH9 71583096 IC50 = 860 nM T27812 CC85VD 71583203 IC50 = 660 nM T27812 C27NXW 71612687 IC50 > 1000 nM T27812 CWZ04H 71612688 IC50 = 6 nM T27812 CJPR13 71625847 Ki = 15.85 nM T27812 C82CJN 71661340 Ki = 2.3 nM T27812 CP7S0W 71661341 Ki = 0.9 nM T27812 COU1K0 71661342 Ki = 24 nM T27812 CM79HR 71661343 Ki = 539 nM T27812 C34LBW 71661346 Ki = 174 nM T27812 C4ZQU3 71661347 Ki = 12 nM T27812 CSWP81 71661348 Ki = 20 nM T27812 CQ2YJ9 71661532 Ki = 212 nM T27812 C1ORE9 71661533 Ki = 12 nM T27812 CBI0U3 71664049 Ki = 8 nM T27812 CZWN24 71716486 IC50 = 31.62 nM T27812 CCI3U0 71717343 Ki = 0.08 nM T27812 CH8O3Z 71717705 IC50 = 6.31 nM T27812 CPA6Y9 71717939 Ki = 1 nM T27812 C0O4ID 71718185 Ki = 31 nM T27812 C7TCH6 71718282 Ki = 392 nM T27812 CF2AW7 71719112 IC50 = 5300 nM T27812 CM7T0H 71719533 IC50 = 0.5012 nM T27812 C2EWG5 71719830 Ki = 230 nM T27812 CMI1V5 71720664 IC50 = 1.7 nM T27812 CY6DR8 71727648 IC50 = 12 nM T27812 CA3H0X 71727754 IC50 = 79 nM T27812 C2WD4V 71727756 IC50 = 16 nM T27812 CDT2P5 71727758 IC50 = 9.1 nM T27812 C39EUA 71727760 IC50 = 9.2 nM T27812 C8BLG9 71727762 IC50 = 340 nM T27812 C1XB7U 71727764 IC50 = 5.2 nM T27812 CS83FB 71727766 IC50 = 9.3 nM T27812 CX7O8K 71727768 IC50 = 11 nM T27812 CEM15Z 71727886 IC50 = 21 nM T27812 C5BL4F 71727888 IC50 = 18 nM T27812 CX21QS 71727890 IC50 = 37 nM T27812 COUT12 71812204 IC50 = 130 nM T27812 CJ7VK8 72202849 IC50 = 3757 nM T27812 CDG0A8 72202852 IC50 = 6451 nM T27812 CV5TJ6 72202983 IC50 = 965.4 nM T27812 CWH6T3 72548703 IC50 = 1.7 nM T27812 C48RGH 72737188 Ki = 71.4 nM T27812 CAEQ04 72737189 Ki = 2.4 nM T27812 C8Q1PJ 72792490 Ki = 3600 nM T27812 CLE86V 72793613 IC50 = 4700 nM T27812 C5KE6Q 72793641 IC50 = 5300 nM T27812 CW1KN9 72793679 IC50 = 4900 nM T27812 CT9YM0 72793681 IC50 = 3000 nM T27812 CZL3M4 72793695 IC50 = 5800 nM T27812 CC65OA 73213195 Ki > 10000 nM T27812 CW83DK 73213196 Ki = 413 nM T27812 C0HTU4 73345764 IC50 = 3530 nM T27812 CESR23 73345847 IC50 = 97 nM T27812 CK48PN 73347369 Ki = 0.75 nM T27812 C4YV6S 73347524 IC50 = 690 nM T27812 CEQS50 73347526 IC50 = 120 nM T27812 CI0JV6 73347528 IC50 = 32 nM T27812 CR97NO 73347825 Ki = 71 nM T27812 CAZ9C2 73348087 IC50 = 57 nM T27812 C85LKM 73348886 Ki = 0.21 nM T27812 C9Y6OD 73348887 Ki = 0.84 nM T27812 CM50LN 73349057 IC50 = 2.1 nM T27812 C7XOF4 73349320 IC50 = 85.6 nM T27812 CW8A0Y 73349359 Ki = 712 nM T27812 CHNT68 73350623 IC50 = 5.7 nM T27812 CCD70L 73353582 IC50 = 180 nM T27812 C1NJ0R 73353884 Ki = 1993 nM T27812 C10ASZ 73355420 Ki > 10000 nM T27812 CN5V0R 73355421 Ki > 10000 nM T27812 CVHQ86 73355688 Ki = 7.3 nM T27812 CWK70C 73356510 Ki = 0.23 nM T27812 C2E7QW 75201901 Ki > 10000 nM T27812 C50CMV 76309752 Ki = 8685 nM T27812 C7O5MI 76311027 IC50 = 970 nM T27812 CRK8G2 76314641 Ki = 8300 nM T27812 CZJH91 76314659 IC50 > 1000 nM T27812 CB5KG6 76314660 IC50 = 190 nM T27812 C1Y9WZ 76316965 Ki = 347 nM T27812 CRMT56 76318226 IC50 > 1000 nM T27812 C62AXF 76318227 IC50 = 150 nM T27812 CJX71S 76320688 Ki = 3010 nM T27812 CR05PL 76322043 IC50 = 420 nM T27812 CQ3CW1 76322044 IC50 = 89 nM T27812 C8YW4N 76324331 Ki = 4180 nM T27812 C3B0YJ 76325557 IC50 = 520 nM T27812 CQJ13A 76325558 IC50 > 1000 nM T27812 CP1U7E 76327897 Ki = 3920 nM T27812 C8S1PB 76327898 Ki = 2640 nM T27812 C1WZ5N 76331540 Ki = 13600 nM T27812 C47EDP 76331541 Ki = 4150 nM T27812 C5N6LG 76331542 Ki = 17200 nM T27812 CN52UF 76332768 IC50 = 250 nM T27812 C0B3HG 76332769 IC50 = 280 nM T27812 C4G6RW 76335160 Ki = 10900 nM T27812 CM54ZS 76335161 Ki = 502 nM T27812 C9ZMB0 76336391 IC50 = 680 nM T27812 C92WBQ 76336500 IC50 = 1218 nM T27812 C28RIZ 76518514 Ki = 414 nM T27812 CP76JG 88912137 Ki = 224 nM T27812 CG1SL7 89723211 IC50 = 740 nM T27812 C2BM9L 89768534 IC50 = 600 nM T27812 CB4Y7R 89768546 IC50 = 520 nM T27812 CP29UR 89838714 IC50 = 120 nM T27812 CF6P3I 89843681 IC50 = 11 nM T27812 C0MX8Y 90645015 Ki = 11 nM T27812 CFB98A 90645017 Ki = 180 nM T27812 C7AX0K 90645019 Ki = 11 nM T27812 CH0VU3 90645021 Ki = 3 nM T27812 C4JOT3 90655117 Ki = 1940 nM T27812 CK3D1X 90655118 Ki = 89 nM T27812 CV4H2G 90655120 Ki = 28 nM T27812 CUJQ70 90655121 Ki = 57 nM T27812 C2P0LK 90655123 Ki > 1000 nM T27812 CVQC46 90655124 Ki > 1000 nM T27812 CBI6Y5 90664323 IC50 = 257 nM T27812 C2PV7O 90664324 IC50 = 33 nM T27812 CO4V5L 90664325 IC50 = 84 nM T27812 C2RW9Y 90664326 IC50 = 76 nM T27812 C6T1KX 90664327 IC50 = 13 nM T27812 C81IBN 90664328 IC50 = 37 nM T27812 C75ZUE 90664329 IC50 = 5 nM T27812 CM7HQ9 90664330 IC50 = 9.17 nM T27812 CA2BO3 90664449 IC50 = 195 nM T27812 C9ULV4 90664450 IC50 = 200 nM T27812 CH02GV 90664451 IC50 = 715 nM T27812 CIL2W9 90664452 IC50 = 181.7 nM T27812 C7RT9G 90664453 IC50 = 12.2 nM T27812 C3AX1O 90664454 IC50 = 447.2 nM T27812 CPGI68 90664459 IC50 = 47 nM T27812 CICD63 90664460 IC50 = 66 nM T27812 CBZT19 90664586 IC50 = 65 nM T27812 C5HRY0 90664587 IC50 = 80 nM T27812 CG6V1D 90664589 IC50 = 13 nM T27812 C7W5SH 90664590 IC50 = 49 nM T27812 CNU6J8 90664598 IC50 = 18 nM T27812 CB95PE 90664599 IC50 = 71.1 nM T27812 CA68PB 90664600 IC50 = 245 nM T27812 C4MUI2 90664601 IC50 = 10.2 nM T27812 CA79EY 90664683 IC50 = 110 nM T27812 CHY82Q 90664697 IC50 = 2.9 nM T27812 CM0Y7P 90664699 IC50 = 84 nM T27812 CEF0R5 90664700 IC50 = 55 nM T27812 CR07QH 90664701 IC50 = 12.4 nM T27812 CZ69VH 90664702 IC50 = 36 nM T27812 CF4P3I 90664703 IC50 = 20 nM T27812 CR7LX6 90664705 IC50 = 51.8 nM T27812 CNT10P 90664709 IC50 = 17 nM T27812 C35BTL 90664710 IC50 = 82 nM T27812 CDPV60 90664712 IC50 = 13 nM T27812 CG7D2H 90664713 IC50 = 35 nM T27812 CZJN57 90664814 IC50 = 1276 nM T27812 CR87PO 90664815 IC50 = 28 nM T27812 CN7W8A 90664816 IC50 = 82 nM T27812 CI8B6Q 90664817 IC50 = 478.4 nM T27812 CEN36Q 90664818 IC50 = 6.17 nM T27812 CJ73WT 90664819 IC50 = 20 nM T27812 C5AWS4 90664820 IC50 = 39.1 nM T27812 CL3AW1 90664821 IC50 = 443 nM T27812 C1C2HB 90664822 IC50 = 3.9 nM T27812 CQ4T3E 90664830 IC50 = 67.2 nM T27812 CTR58M 90664931 IC50 = 397 nM T27812 CP9SI1 90664949 IC50 = 42 nM T27812 CZ19LO 90664951 IC50 = 10.2 nM T27812 CLN9K2 90664952 IC50 = 39 nM T27812 CO5Y3C 90664958 IC50 = 7.3 nM T27812 C74XDT 90664959 IC50 = 2.7 nM T27812 CWQ18M 90664960 IC50 = 6.2 nM T27812 C07WIP 90664961 IC50 = 370 nM T27812 CHT7D5 90664962 IC50 = 129 nM T27812 C04UEP 90665072 IC50 = 347 nM T27812 CF90MU 90665073 IC50 = 9.1 nM T27812 C8YX4R 90665074 IC50 = 281.9 nM T27812 CP5QO8 90665075 IC50 = 232 nM T27812 C3XIQ2 90665076 IC50 = 9.53 nM T27812 CI8JU1 90665077 IC50 = 16.8 nM T27812 C67AXN 90665078 IC50 = 25 nM T27812 CQ95OT 90665079 IC50 = 24 nM T27812 C7JLM9 90665080 IC50 = 17 nM T27812 CZHA09 90665086 IC50 = 4.88 nM T27812 C17EWV 90665087 IC50 = 14 nM T27812 CO46PW 90665091 IC50 = 18 nM T27812 CXJ62T 90665173 IC50 = 28 nM T27812 CYD25E 90665193 IC50 = 12 nM T27812 CG98QO 90665194 IC50 = 17.8 nM T27812 C5PN4D 90665195 IC50 = 14.2 nM T27812 C7XIS2 90665197 IC50 = 19 nM T27812 CIJ5M0 90665200 IC50 = 28 nM T27812 C09JPN 90665201 IC50 = 106 nM T27812 C8BV5P 90665202 IC50 = 15.8 nM T27812 CBH87U 91667621 IC50 = 84 nM T27812 C0RV4M 91799659 IC50 = 83 nM T27812 C0XJT5 118626089 Ki = 76 nM T27812 CA79GZ 118706038 IC50 = 73.8 nM T27812 CGBC58 118706039 IC50 = 83.4 nM T27812 C5LCJ1 118706532 IC50 = 71.9 nM T27812 CI2FN5 118706536 IC50 = 51.3 nM T27812 C2BG1F 118706537 IC50 = 47.1 nM T27812 C2WP6X 118706538 IC50 = 46.3 nM T27812 CZE4U0 118706539 IC50 = 36.6 nM T27812 CX8I0G 118706540 IC50 = 58.1 nM T27812 C4S9VT 118706541 IC50 = 37.5 nM T27812 CKD94F 118706542 IC50 = 37.7 nM T27812 C0KQO9 118706543 IC50 = 23 nM T27812 C5HJY0 118706544 IC50 = 38.5 nM T27812 CJ15AS 118708361 IC50 = 50 nM T27812 C7XEC0 118708362 IC50 = 2200 nM T27812 CK30WF 118708364 IC50 = 1300 nM T27812 CG7W4D 118708365 IC50 = 1900 nM T27812 C6UJC5 118708366 IC50 = 4300 nM T27812 CLQ52I 118708373 IC50 = 260 nM T27812 CSB25E 118709750 Ki = 227 nM T27812 CD4S9R 118709751 Ki = 102 nM T27812 CD34IY 118710582 IC50 = 3 nM T27812 CD1O7G 118710583 IC50 = 2500 nM T27812 C5GRY0 118713756 IC50 = 6.2 nM T27812 C4VAE0 118713757 IC50 = 333 nM T27812 CPDB78 118713768 IC50 = 23 nM T27812 C84GOU 118713773 IC50 = 114 nM T27812 CW0SN9 118713774 IC50 = 87.9 nM T27812 CUN71K 118713775 IC50 = 14.6 nM T27812 C6ZL1K 118713793 IC50 = 44.8 nM T27812 CQFH60 118713795 IC50 = 34 nM T27812 CC58ZS 118713797 IC50 = 11.4 nM T27812 C2LY9D 118713799 IC50 = 11.1 nM T27812 CMO2V7 118713801 IC50 = 7.6 nM T27812 C9LKI0 118713803 IC50 = 42.2 nM T27812 CD2C1A 118713804 IC50 = 20.2 nM T27812 C2OZ7H 118713805 IC50 = 179 nM T27812 CM4P8X 118713806 IC50 = 99.9 nM T27812 C7EXQ9 118713807 IC50 = 1.6 nM T27812 C05FSJ 118714012 IC50 = 621.3 nM T27812 CU59IA 118714013 IC50 = 905.3 nM T27812 CGC5J6 118719847 IC50 = 2200 nM T27812 C6HV3B 118730351 EC50 > 10000 nM T27812 C3LZM9 118730352 IC50 > 10 nM T27812 CDU18K 118871456 IC50 = 436100 nM T27812 CU4CW1 121313969 IC50 = 10400 nM T27812 CSC5J4 121488665 Ki = 15.8 nM T27812 CS7K8R 122180523 Ki = 227 nM T27812 CJ56CG 122180524 Ki = 38 nM T27812 CR7PD6 122180525 Ki = 24 nM T27812 CUK9E2 122181877 IC50 = 480 nM T27812 CHKY46 122181879 IC50 = 680 nM T27812 CR5ES2 122188495 IC50 = 422 nM T27812 C5Y2LX 122188496 IC50 = 546 nM T27812 CG6UW3 122188497 IC50 = 500 nM T27812 C12TIS 122188498 IC50 = 449 nM T27812 CL7PH5 122188499 IC50 = 56 nM T27812 C9TDA7 122188500 IC50 = 7670 nM T27812 CARF60 122188503 IC50 = 100 nM T27812 CC87DN 122188504 IC50 = 1914 nM T27812 CQZ0A3 122188505 IC50 = 323 nM T27812 CHVR64 122188579 Ki < 10000 nM T27812 C8L1FV 122188773 IC50 = 986 nM T27812 CJ6G5D 122188774 IC50 > 10000 nM T27812 CNT50I 122188775 IC50 > 10000 nM T27812 CA8QW0 122188776 IC50 = 786 nM T27812 C3VDY7 122197403 Ki = 1.3 nM T27812 C1MFJ3 122197404 Ki = 8.8 nM T27812 C7GO0U 122197405 Ki = 1.3 nM T27812 CTBN56 127026052 Ki = 36.31 nM T27812 C4D9QY 127026491 IC50 = 800 nM T27812 C8MC1I 127028408 Ki = 1258.93 nM T27812 CEJ3R5 127029340 IC50 = 18 nM T27812 C6H5KN 127030249 IC50 = 4320 nM T27812 CCD8P5 127032017 IC50 = 4920 nM T27812 CQS75W 127032626 IC50 = 2000 nM T27812 CX6J8Y 127033284 IC50 = 2030 nM T27812 CY82JA 127033285 IC50 = 2250 nM T27812 CU8K1Q 127033286 IC50 = 1460 nM T27812 C1ZMH0 127033287 IC50 = 2610 nM T27812 C0YF3E 127033288 IC50 = 2510 nM T27812 C3IPX2 127033888 IC50 = 1360 nM T27812 CF3XL5 127033889 IC50 = 1760 nM T27812 C5QGV3 127033890 IC50 = 1180 nM T27812 CR61YN 127034912 Ki < 100 nM T27812 CQ0ZT9 127035062 Ki = 1001 nM T27812 CU49VE 127036186 Ki = 363.08 nM T27812 CG06BD 127036932 Ki = 40.74 nM T27812 CVW71O 127036953 Ki = 125.89 nM T27812 C7L1DB 127037832 IC50 > 10000 nM T27812 CG0VP9 127046067 IC50 = 940 nM T27812 CLR5B3 127046068 IC50 = 300 nM T27812 CL80OZ 127046276 IC50 = 420 nM T27812 CE6CI9 127046277 Ki = 500 nM T27812 C61QFA 127046278 Ki = 1600 nM T27812 C6ZW0O 127046826 IC50 = 600 nM T27812 C78LAW 127046946 Ki = 280 nM T27812 C2AG0M 127046947 IC50 = 350 nM T27812 C6KV1C 127046964 IC50 = 280 nM T27812 C52KRU 127046965 IC50 = 270 nM T27812 C9AUY1 127046966 Ki = 640 nM T27812 C51UDC 127046967 Ki = 35 nM T27812 C1I8VZ 127047091 Ki = 1800 nM T27812 C5U3XA 127047092 IC50 = 440 nM T27812 CUDG72 127047515 Ki = 2800 nM T27812 CJAX61 127047516 Ki = 290 nM T27812 CU0MX9 127047629 Ki = 27 nM T27812 CN3R2W 127047781 Ki = 270 nM T27812 C42FHY 127049060 Ki = 4.677 nM T27812 C6HJ5B 127049763 IC50 = 24 nM T27812 C51TDU 127049764 IC50 = 5 nM T27812 CL59OV 127050294 IC50 = 11 nM T27812 CX53AC 127050632 Ki = 3056 nM T27812 C6Q7TA 127051504 IC50 = 29 nM T27812 CTL8J1 127051843 Ki = 895 nM T27812 C8TNB1 127051845 Ki = 2442 nM T27812 C5ONG1 127051864 Ki = 180 nM T27812 CVQW26 127051865 Ki = 4.677 nM T27812 CWJ59Z 127051882 IC50 = 730 nM T27812 CCY71I 127052465 Ki > 10000 nM T27812 C2E9VX 127052467 Ki = 113 nM T27812 CPO4C3 127052468 Ki = 163 nM T27812 CSQ2N8 127052486 Ki = 386 nM T27812 C4YJ8H 127052487 Ki = 25 nM T27812 CLU7C1 127052757 Ki = 4284 nM T27812 C50GOC 130442480 Ki > 10000 nM T27812 CM04RF 130442572 Ki = 9700 nM T27812 C1RI8Q 132060720 Ki = 2477 nM T27812 CY8B9L 132060743 Ki = 1376 nM T27812 CXV95T 132578504 IC50 > 10000 nM T27812 C8NUR9 132578505 IC50 > 10000 nM T27812 CGW0I7 132578506 IC50 > 10000 nM T27812 C5GEB2 132578508 IC50 > 10000 nM T27812 CAVB41 132584404 Ki > 10000 nM T27812 C2V8BH 134133118 Ki = 28 nM T27812 C3P9IJ 134136137 Ki = 32.7 nM T27812 CLA4R3 134136207 Ki = 102 nM T27812 C7L2SN 134136382 Ki = 274 nM T27812 C3F8OJ 134137742 Ki = 800 nM T27812 CSIQ62 134140156 Ki = 11000 nM T27812 C8TC3Z 134140440 Ki = 25.6 nM T27812 CWQG03 134145252 Ki = 37.5 nM T27812 CK37OV 134145259 Ki = 30.5 nM T27812 CLUV50 134145912 Ki = 65.3 nM T27812 CL9RW7 134148069 Ki = 18.9 nM T27812 CBU81N 134149168 Ki > 10000 nM T27812 CA50EU 134150000 Ki = 212 nM T27812 CHK9J1 134150839 Ki = 26.9 nM T27812 C5SK4P 134154831 Ki = 14 nM T27812 C43MXR 134155275 Ki = 14000 nM T27812 CU3S0L 134156929 Ki < 100 nM T27812 C1GY2T 135156251 EC50 > 10000 nM T27812 CKO6D5 135405894 Ki = 154 nM T27812 C7HYA8 135440165 Ki = 8.9 nM T27812 CMK06P 135477797 Ki = 15 nM T27812 C1IKQ6 135499867 Ki = 84 nM T27812 CTP2R6 135519400 Ki = 3.6 nM T27812 CA39PK 135519421 Ki = 151 nM T27812 CCBM21 135545454 Ki = 9.7 nM T27812 C5J9BC 136019934 Ki = 8.9 nM T27812 CXA5Y9 136044137 Ki = 1.5 nM T27812 C0TAI6 136274356 Ki = 22 nM T27812 CF7S1X 136274357 Ki = 0.5 nM T27812 C3QOP1 136340699 IC50 = 380 nM T27812 C4UON5 136389176 IC50 = 120 nM T27812 CG05IL 136389183 IC50 > 1000 nM T27812 CP0E8J 136389204 IC50 > 1000 nM T27812 C48SIG 137628671 Ki = 750 nM T27812 C3USH9 137631428 Ki < 10000 nM T27812 C2QCA5 137631487 IC50 > 10000 nM T27812 C5XL1N 137631893 Ki = 1.27 nM T27812 C14RKA 137632704 IC50 = 120500 nM T27812 C0C6ZL 137632750 IC50 = 1240 nM T27812 CI69VT 137633306 Ki < 10000 nM T27812 C5G0XW 137633601 IC50 > 10 nM T27812 C9P2KQ 137634088 IC50 = 2300 nM T27812 C8HPN4 137634334 IC50 > 10000 nM T27812 C2LJW0 137634948 IC50 = 3960 nM T27812 CR74SC 137635327 IC50 = 8000 nM T27812 CW9X5R 137635426 IC50 = 7500 nM T27812 CX17BR 137635648 IC50 = 880 nM T27812 C94VXJ 137635884 Ki = 5.4 nM T27812 C42HCS 137636472 IC50 = 5000 nM T27812 CK68DP 137636508 IC50 = 8 nM T27812 CKQ92P 137636703 IC50 = 2000 nM T27812 COH18X 137637663 IC50 = 118400 nM T27812 CL56ZQ 137637671 IC50 > 10000 nM T27812 CD31YG 137638231 IC50 = 310 nM T27812 C1EU5S 137638283 IC50 = 5250 nM T27812 CJI0K6 137638828 IC50 > 10 nM T27812 CBK0I8 137639266 IC50 > 10 nM T27812 CI5Q2P 137639497 Ki < 10000 nM T27812 C3FSN5 137639697 IC50 = 10 nM T27812 CGB0E4 137640270 IC50 = 1100 nM T27812 CV20BW 137640543 IC50 = 1670 nM T27812 CVC6R8 137640624 IC50 > 10000 nM T27812 C3C1XS 137640629 IC50 = 2400 nM T27812 C1X0QZ 137640906 IC50 = 3130 nM T27812 C06KGS 137641034 IC50 = 4050 nM T27812 CE8N4S 137641762 Ki = 3100 nM T27812 CKS5V0 137643541 Ki < 10000 nM T27812 C70XZQ 137643636 IC50 > 10000 nM T27812 C9VR5M 137643839 IC50 = 4960 nM T27812 CASM14 137643954 IC50 = 59600 nM T27812 CV85OM 137644057 EC50 = 38000 nM T27812 CTFI60 137644452 Ki = 5600 nM T27812 C3ZRY2 137645338 IC50 = 8810 nM T27812 CPCY48 137645406 Ki = 295 nM T27812 C6LQZ0 137645491 Ki < 10000 nM T27812 COES67 137645514 Ki < 10000 nM T27812 C85OYG 137645602 IC50 = 158.7 nM T27812 C1KT5F 137645761 IC50 > 10000 nM T27812 CPZ3E1 137646230 IC50 = 8000 nM T27812 CN4T3X 137646510 EC50 = 1600 nM T27812 CE9M3Z 137648195 IC50 = 3910 nM T27812 CIH3O8 137648265 IC50 = 4830 nM T27812 CL06NY 137648464 IC50 > 10000 nM T27812 C0EVB7 137648614 IC50 = 6290 nM T27812 CG1ME5 137648669 IC50 = 1320 nM T27812 CUFO39 137649223 IC50 = 8794 nM T27812 CO2YH7 137649677 IC50 = 70900 nM T27812 C6YE5R 137649990 IC50 = 44700 nM T27812 C37GZJ 137651008 Ki < 10000 nM T27812 CWG87E 137651507 Ki < 10000 nM T27812 CU4S1W 137651887 Ki = 6.2 nM T27812 C6GL0F 137652257 IC50 = 5050 nM T27812 C65XKJ 137653127 IC50 > 10000 nM T27812 CR9F3Q 137653203 Ki < 10000 nM T27812 C02HUF 137653618 IC50 > 10000 nM T27812 CR25WM 137653998 Ki < 10000 nM T27812 C1JGO6 137654323 IC50 > 10000 nM T27812 CT35OC 137654501 IC50 = 5130 nM T27812 C96BJN 137654642 IC50 = 6910 nM T27812 C46UFA 137654647 IC50 = 4050 nM T27812 CX82HS 137654666 Ki = 2.6 nM T27812 C8FWX6 137654918 IC50 = 280 nM T27812 CL41SG 137655166 EC50 = 31000 nM T27812 CF7M8V 137655321 IC50 = 3860 nM T27812 C3LG7W 137655838 IC50 > 10000 nM T27812 CU3DK5 137655842 IC50 = 7700 nM T27812 CG8TW9 137656204 Ki < 10000 nM T27812 CZ84KG 137656433 IC50 = 1500 nM T27812 CN2UE9 137656598 IC50 > 10000 nM T27812 CQ1SI8 137656684 IC50 = 1414 nM T27812 CZ1XS0 137656786 IC50 = 57200 nM T27812 C56MCJ 137656979 Ki < 10000 nM T27812 C3GX2Z 137657462 IC50 = 209500 nM T27812 CML7S0 137658465 Ki < 10000 nM T27812 COV16Y 137659590 IC50 = 190 nM T27812 CG92PT 137660066 IC50 = 550 nM T27812 CWX6N4 137660247 IC50 = 540 nM T27812 CEV40N 137661034 IC50 > 10000 nM T27812 CLF7V1 137661266 IC50 = 5220 nM T27812 C28EJN 137661323 Ki < 10000 nM T27812 CCSU34 137661732 IC50 = 1350 nM T27812 C4VP7A 137662010 IC50 = 160 nM T27812 CS47KN 137662116 IC50 = 1121 nM T27812 C4E5ZX 141363479 IC50 > 10000 nM T27812 COT18S 145011254 Ki > 10000 nM T27812 CG8ZX0 145960719 IC50 = 314.1 nM T27812 CQR07X 145960843 IC50 = 20.42 nM T27812 CP2M6G 145961773 IC50 = 22.1 nM T27812 C2A3DR 145962768 IC50 = 229.3 nM T27812 C9A1VD 145967813 IC50 = 11 nM T27812 C76SHX 145968149 Ki = 202 nM T27812 C3DZ7P 145968324 Ki = 1.41 nM T27812 C3D0LR 145968390 Ki = 2.59 nM T27812 CT09GI 145968506 Ki = 9.85 nM T27812 CM8TF3 145968603 Ki = 31.62 nM T27812 C9S8QE 145968791 Ki = 18.5 nM T27812 CM0Z9G 145968895 Ki = 111 nM T27812 CVU49S 145969204 Ki = 5.4 nM T27812 CERC65 145969459 Ki = 246 nM T27812 CD3Z4I 145969495 Ki = 14.1 nM T27812 C4BS6T 145969809 IC50 = 0.72 nM T27812 C3FNX8 145969978 Ki = 2.39 nM T27812 CUQ7E0 145970103 Ki = 0.3162 nM T27812 CRZN24 145970238 Ki = 5.47 nM T27812 CBT6L8 145970391 IC50 = 10 nM T27812 CF67IA 145970695 Ki = 5.012 nM T27812 C6FBU7 145970863 Ki = 1.74 nM T27812 CB7O9W 145971077 Ki = 63.1 nM T27812 CT5CX0 145973771 Ki = 2080 nM T27812 C90NFP 145976326 Ki = 195.02 nM T27812 CS4FG0 145979497 Ki = 0.16 nM T27812 C87MSW 145980271 Ki = 10000 nM T27812 CVKQ04 145981108 IC50 = 3150 nM T27812 CV1J4B 145981842 IC50 = 2800 nM T27812 C2A7WP 145982315 IC50 = 680 nM T27812 CE0CB8 145983354 IC50 > 10000 nM T27812 CE84XH 145983742 IC50 = 741.4 nM T27812 CO45RG 145983783 IC50 = 1320 nM T27812 C8F0IL 145983986 IC50 = 230 nM T27812 CU53SY 145984002 IC50 > 10000 nM T27812 C9ZRP0 145984032 IC50 = 273 nM T27812 CU6QS4 145984074 IC50 > 10000 nM T27812 CJ9UZ0 145984374 IC50 > 10000 nM T27812 C6I3NT 145984803 IC50 = 4270 nM T27812 C7EIC6 145984821 IC50 = 6850 nM T27812 C6M1FI 145984939 IC50 = 400 nM T27812 C9W6PO 145984940 IC50 > 10000 nM T27812 CT6KH5 145985061 IC50 = 740 nM T27812 C8KUD1 145985187 Ki = 487 nM T27812 CG2C8H 145985476 IC50 = 6940 nM T27812 C82KFY 145985630 IC50 = 1080 nM T27812 C1WA5L 145985747 IC50 = 550 nM T27812 C1H2UT 145985812 IC50 = 9640 nM T27812 C5XC2O 145986024 IC50 = 1010 nM T27812 C5XCV8 145986058 IC50 = 1170 nM T27812 CG0Q1F 145986130 IC50 = 460 nM T27812 CG86VQ 145986485 Ki = 10.7 nM T27812 COT25D 145986575 Ki = 74.6 nM T27812 CNJH37 145986752 Ki = 1314 nM T27812 CUGO10 145988693 Ki = 903 nM T27812 CW6E8Z 145989332 IC50 = 5160 nM T27812 CB6OP0 145989720 Ki = 0.41 nM T27812 C0X7BO 145990773 IC50 = 990 nM T27812 CNBS32 145991101 IC50 = 1860 nM T27812 C5K3CS 145991656 IC50 = 830 nM T27812 CBZY16 145993315 IC50 = 4320 nM T27812 CZP9L5 145993640 IC50 = 10700 nM T27812 CGTV18 145994198 IC50 = 1040 nM T27812 CC2G1V 146025727 Ki > 10000 nM T27812 C1Z7ED 155513346 IC50 > 10000 nM T27812 CH4Z9J 155513656 IC50 = 29700 nM T27812 CJ87WT 155514907 IC50 > 10000 nM T27812 CCF56N 155515030 IC50 = 144600 nM T27812 CB71XT 155517422 IC50 = 264400 nM T27812 CRM7H5 155521227 IC50 > 10000 nM T27812 CZLF49 155521764 IC50 > 10000 nM T27812 CAFT73 155522329 Ki = 111 nM T27812 C5KYB4 155524228 Ki = 201 nM T27812 C7F2ZG 155524366 Ki = 63 nM T27812 CWD38V 155524413 IC50 > 10000 nM T27812 CVF9H3 155524550 IC50 > 10000 nM T27812 CVF9E8 155525067 IC50 = 201500 nM T27812 CHJ79N 155528236 Ki = 221 nM T27812 CFMJ93 155528557 IC50 = 24700 nM T27812 CVNK03 155529810 IC50 = 140000 nM T27812 C2JVS7 155530463 IC50 = 15800 nM T27812 C2MB4H 155533557 IC50 > 10000 nM T27812 CSE59K 155534331 Ki = 140 nM T27812 C8R2TB 155534729 Ki = 150.5 nM T27812 C35NRU 155535386 Ki = 314 nM T27812 C0WX1T 155535629 IC50 > 10000 nM T27812 CRHA67 155536435 IC50 = 58650 nM T27812 CAT98F 155539483 Ki = 32.4 nM T27812 CV9KY1 155539925 Ki = 523 nM T27812 CNU92V 155540807 Ki = 705 nM T27812 C4STU5 155543525 Ki > 10000 nM T27812 C0QN3W 155543949 Ki = 141.8 nM T27812 CE5YV0 155545747 IC50 > 10000 nM T27812 C1URC8 155547273 Ki = 2946 nM T27812 C2KM3J 155547346 IC50 = 76.3 nM T27812 CLH68U 155549829 IC50 > 10000 nM T27812 CAS6B5 155550042 Ki > 10000 nM T27812 C0UYA7 155551050 IC50 = 200800 nM T27812 C1U2KX 155554780 IC50 > 10000 nM T27812 CXM7C6 155555638 Ki = 30 nM T27812 CH6ZD0 155556044 IC50 > 10000 nM T27812 C4AG0H 155558726 IC50 > 100000 nM T27812 C5B2OZ 155559232 Ki > 10000 nM T27812 C28MCV 155559835 Ki > 10000 nM T27812 C4O8LX 155560376 IC50 = 220900 nM T27812 CU6YD0 155560597 IC50 = 362800 nM T27812 C5AI0S 155562519 Ki = 17.5 nM T27812 CRCW25 155562997 Ki = 51 nM T27812 CV9O7W 155563205 Ki = 1313 nM T27812 CR12DI 155565189 Ki = 3400 nM T27812 C0D8ZO 155566396 Ki = 156 nM T27812 C4EX7C 155568246 Ki = 308 nM T27812 CV5H3F 155568689 Ki = 102 nM T27812 C3N9VU 10251906 Ki > 500 nM T27812 CP9TR0 10324985 Ki = 6144 nM T27812 CB2VD8 44241743 Ki = 61 nM T27812 CUKM52 44586281 Ki = 11.4 nM T27812 CNG2T7 44586282 Ki = 1910 nM T27812 CP9ED8 44586283 Ki = 374 nM T27812 COY7T4 44586284 Ki = 213 nM T27812 D00DDT 46882974 EC50 = 28840.32 nM T27812 D00DEH 45483512 EC50 = 186 nM T27812 D00EUD 43565977 EC50 = 17579.24 nM T27812 D00FMX 46230706 Ki = 292 nM T27812 D00GDI 45487890 Ki = 1480 nM T27812 D00HCC 12996705 Ki = 1880 nM T27812 D00KRQ 23113096 Ki = 1760 nM T27812 D00QCP 46837647 IC50 > 100000 nM T27812 D00RTM 52549 IC50 = 58 nM T27812 D00WMS 3047299 Ki > 10000 nM T27812 D01ABR 44414723 Ki = 18 nM T27812 D01AOI 44592200 IC50 = 15 nM T27812 D01CXD 10398175 Ki > 10000 nM T27812 D01EIS 12263801 IC50 = 14 nM T27812 D01FFX 24691160 IC50 = 8 nM T27812 D01GSG 44592199 IC50 = 42 nM T27812 D01JYY 11323940 IC50 = 5 nM T27812 D01KAX 135453290 Ki > 10000 nM T27812 D01MBF 45483536 Ki = 157 nM T27812 D01RWY 44542656 Ki > 10000 nM T27812 D01SHR 44593693 IC50 = 2100 nM T27812 D01WWC 16573 Ki > 950 nM T27812 D01YED 45141808 IC50 > 100 nM T27812 D01YNZ 45483529 Ki = 74 nM T27812 D02BXA 238317 Ki > 10000 nM T27812 D02DCM 44230874 Ki = 15 nM T27812 D02EKR 3031077 Ki > 10000 nM T27812 D02ENH 9797657 IC50 = 13 nM T27812 D02ICX 14373 IC50 = 2780 nM T27812 D02JVG 44399737 EC50 < 10000 nM T27812 D02LQG 170832 Ki = 182 nM T27812 D02MMS 44613577 EC50 = 257039.58 nM T27812 D02NUR 44543266 Ki > 10000 nM T27812 D02TMK 1614 IC50 = 478 nM T27812 D02VHZ 44613455 EC50 = 5888.44 nM T27812 D02YOO 4500 Ki = 1.4 nM T27812 D02YSN 11651575 IC50 = 636 nM T27812 D02ZIQ 43227131 IC50 = 970 nM T27812 D03BQV 3033806 IC50 = 320 nM T27812 D03DQQ 45375938 EC50 = 915 nM T27812 D03EMO 16102754 IC50 = 1500 nM T27812 D03ETK 44613192 EC50 = 39810.72 nM T27812 D03FGM 44414732 IC50 = 210 nM T27812 D03HFH 46882993 EC50 = 3715.35 nM T27812 D03HQF 11644566 IC50 = 50 nM T27812 D03JOX 11311147 IC50 = 2020 nM T27812 D03MYV 44414735 IC50 = 87 nM T27812 D03XMD 11983346 Ki = 25.12 nM T27812 D03YQY 46837650 IC50 > 100000 nM T27812 D03ZDY 44414750 IC50 = 15 nM T27812 D04GHK 44613690 EC50 = 10471.29 nM T27812 D04IZU 44568213 IC50 = 60 nM T27812 D04KZX 44542809 IC50 = 790 nM T27812 D04NDO 45483400 Ki = 56 nM T27812 D04NKQ 22599992 Ki = 319 nM T27812 D04RUF 44613456 EC50 = 61235.04 nM T27812 D04ZPF 45483409 Ki = 26 nM T27812 D05FMK 44613068 EC50 = 23988.33 nM T27812 D05GDP 599482 Ki > 10000 nM T27812 D05LJC 45483405 Ki = 2970 nM T27812 D05LKO 44414722 Ki = 2 nM T27812 D05LLP 44613453 EC50 = 25703.96 nM T27812 D05PLF 3031066 IC50 = 9800 nM T27812 D05REQ 22139473 IC50 = 32 nM T27812 D05UHO 44613452 EC50 = 16595.87 nM T27812 D05UMA 10334821 Ki = 2.5 nM T27812 D05YHP 44613580 EC50 = 18879.91 nM T27812 D05ZUX 44207909 Ki >= 1000 nM T27812 D06EMC 11392888 Ki = 6 nM T27812 D06KNV 3703 Ki = 0.1995 nM T27812 D06LCK 45141805 IC50 > 100 nM T27812 D06PJD 44593439 IC50 = 327 nM T27812 D06QGD 11357862 IC50 = 1110 nM T27812 D06QIQ 44592241 IC50 = 3 nM T27812 D06UDU 45483520 Ki = 427 nM T27812 D06WIV 44578367 Ki = 1070 nM T27812 D07DMN 44430859 IC50 = 3.1 nM T27812 D07DWS 45483446 Ki = 978 nM T27812 D07IOX 44543268 Ki > 10000 nM T27812 D07LFR 44231007 Ki = 7 nM T27812 D07OOI 3456 IC50 = 289 nM T27812 D07PAT 16102753 IC50 = 3300 nM T27812 D07SAA 44543271 IC50 = 3180 nM T27812 D07SZF 44613576 EC50 = 20941.12 nM T27812 D07TEJ 44414874 IC50 = 38 nM T27812 D07ZOP 11470616 IC50 = 4400 nM T27812 D08AWN 3058751 IC50 = 46 nM T27812 D08BCF 5011 Ki = 30 nM T27812 D08EKQ 46890532 Ki = 15 nM T27812 D08JCK 16102777 Ki = 7800 nM T27812 D08JLB 45483406 Ki = 28 nM T27812 D08LAY 13904719 IC50 = 25 nM T27812 D08MEN 14014889 IC50 = 7800 nM T27812 D08NZE 126280 Ki = 4.8 nM T27812 D08RCH 44566054 IC50 = 3500 nM T27812 D08SCH 151900 IC50 = 74 nM T27812 D08SLZ 16102764 IC50 = 180 nM T27812 D09BYB 45487941 IC50 > 100 nM T27812 D09DWM 44411213 Ki = 0.99 nM T27812 D09FIC 46890395 Ki = 6 nM T27812 D09HJL 10331436 Ki > 10000 nM T27812 D09HLX 39484 Ki = 48000 nM T27812 D09IIH 45483459 EC50 = 1760 nM T27812 D09JRN 44414721 IC50 = 4 nM T27812 D09PIN 3378093 IC50 = 4700 nM T27812 D09QZM 11637187 IC50 = 4 nM T27812 D09RPR 16737207 Ki > 10000 nM T27812 D09VTJ 441298 IC50 = 2000 nM T27812 D09XWL 45141379 IC50 > 100 nM T27812 D09YHS 44613329 EC50 = 2511.89 nM T27812 D0A1HH 44414708 IC50 = 12 nM T27812 D0A3YK 44414860 IC50 = 17 nM T27812 D0A7GW 45487772 IC50 = 28.3 nM T27812 D0A9QT 44456154 Ki = 3.7 nM T27812 D0B4FN 11148955 Ki > 10000 nM T27812 D0B5AG 44560576 IC50 > 10000 nM T27812 D0BM0M 44454695 IC50 > 10000 nM T27812 D0BW0V 44589528 Ki = 9 nM T27812 D0C0GL 3031062 IC50 > 100 nM T27812 D0C5GF 6918515 Ki = 4700 nM T27812 D0CG2Y 44133490 Ki = 1890 nM T27812 D0CK9K 6918513 Ki > 10000 nM T27812 D0D2WN 44613575 EC50 = 46773.51 nM T27812 D0D3QE 11550626 Ki > 10000 nM T27812 D0D5QV 9838803 IC50 = 4600 nM T27812 D0D8YY 44411431 Ki = 8.4 nM T27812 D0E3DM 44592118 IC50 = 23 nM T27812 D0E6PQ 45483451 Ki = 706 nM T27812 D0EO5P 44414709 IC50 = 16 nM T27812 D0EX2M 44414720 IC50 = 9.4 nM T27812 D0F5AQ 49798218 Ki = 3.981 nM T27812 D0F6GB 44133853 Ki = 57 nM T27812 D0FU5E 10220053 Ki = 77 nM T27812 D0G0CJ 45141380 IC50 > 100 nM T27812 D0G1XP 44543273 Ki = 842 nM T27812 D0G5RH 44462219 Ki = 178 nM T27812 D0G6BJ 24802842 Ki = 0.631 nM T27812 D0G8CV 9954003 Ki = 0.2512 nM T27812 D0G8UA 46890321 Ki = 8 nM T27812 D0GG2J 46890492 Ki = 21 nM T27812 D0GY8R 45141807 IC50 > 100 nM T27812 D0H2TS 45483528 Ki = 49 nM T27812 D0H4AD 44542509 IC50 = 2520 nM T27812 D0H7PI 44613579 EC50 = 20892.96 nM T27812 D0HF1N 458519 EC50 = 2118 nM T27812 D0I2UC 44230733 Ki = 4 nM T27812 D0I4TO 10107888 Ki = 18 nM T27812 D0I9KV 11220599 Ki = 830 nM T27812 D0IB6Y 11658526 IC50 = 617 nM T27812 D0IC4J 45375937 Ki = 901 nM T27812 D0IR0R 16102751 IC50 = 1300 nM T27812 D0J4CB 24803184 Ki = 0.1259 nM T27812 D0J5AR 11672904 IC50 = 2260 nM T27812 D0J5EF 215051 IC50 > 100 nM T27812 D0J6JT 1355 Ki = 271 nM T27812 D0J8DC 44414861 IC50 = 12 nM T27812 D0K3EW 49799108 Ki = 0.1259 nM T27812 D0K6ZT 44133851 Ki = 728 nM T27812 D0KD9M 44592198 IC50 = 37 nM T27812 D0KT2M 44133674 Ki = 610 nM T27812 D0L0AY 11506691 Ki = 68 nM T27812 D0L5MW 181743 Ki = 244 nM T27812 D0L6RY 11322641 Ki > 10000 nM T27812 D0L7BK 44414856 IC50 = 23 nM T27812 D0M3TK 45483431 Ki = 994 nM T27812 D0N0TQ 11571886 Ki = 43 nM T27812 D0N2KU 44517677 Ki = 224 nM T27812 D0N2RJ 45483432 Ki = 3100 nM T27812 D0NC3P 117443 IC50 > 200000 nM T27812 D0NM1F 45487774 IC50 = 15 nM T27812 D0NY4W 11152502 IC50 = 197 nM T27812 D0O2LC 44543272 IC50 > 100 nM T27812 D0O8QM 44613067 EC50 = 17378.01 nM T27812 D0O9BL 11210506 IC50 = 1070 nM T27812 D0P6SY 14595987 IC50 = 190 nM T27812 D0P9EO 45141381 IC50 > 100 nM T27812 D0PN9R 16655023 Ki = 1.2 nM T27812 D0Q3EJ 44613458 EC50 = 15135.61 nM T27812 D0Q6SH 45483408 Ki = 2 nM T27812 D0Q8IQ 43794735 IC50 > 100 nM T27812 D0R1AE 44332186 IC50 = 10 nM T27812 D0R3GW 10296414 Ki = 6.31 nM T27812 D0R3TA 45483407 Ki = 274 nM T27812 D0R5AD 43227726 Ki > 10000 nM T27812 D0R7ZC 31721 EC50 = 32359.37 nM T27812 D0R8EV 3027752 Ki > 10000 nM T27812 D0R8TH 16102750 IC50 = 2400 nM T27812 D0R8XV 44613451 EC50 = 19498.45 nM T27812 D0RT9B 11506733 IC50 = 32 nM T27812 D0S1XC 25224941 IC50 = 16 nM T27812 D0S4JT 45483466 Ki = 780 nM T27812 D0S9AY 44592244 IC50 = 11 nM T27812 D0S9IO 44454825 IC50 = 1600 nM T27812 D0SA1G 21978439 EC50 = 12589.25 nM T27812 D0SD4O 46882957 EC50 = 16982.44 nM T27812 D0SN6R 44592197 IC50 = 25 nM T27812 D0SP2J 10257 IC50 = 1200 nM T27812 D0T2RY 9948320 Ki >= 1000 nM T27812 D0T5VG 11514389 Ki = 18 nM T27812 D0T7VU 44613578 EC50 = 21379.62 nM T27812 D0T8BU 13904714 IC50 = 9.5 nM T27812 D0U3SB 45141806 IC50 > 100 nM T27812 D0U7OD 16043230 Ki = 10 nM T27812 D0V0PR 45483527 Ki = 364 nM T27812 D0V5GB 11637190 Ki = 83.18 nM T27812 D0V8IZ 44543267 Ki > 10000 nM T27812 D0VC1K 826600 IC50 = 660 nM T27812 D0VX1V 44613193 EC50 = 28183.83 nM T27812 D0VY9K 45141809 IC50 > 100 nM T27812 D0W6WL 44414840 IC50 = 23 nM T27812 D0W8BJ 44560674 IC50 = 10000 nM T27812 D0W8YO 46230654 EC50 = 915 nM T27812 D0W9JK 11220185 IC50 = 3 nM T27812 D0WB6P 46227262 IC50 = 6.8 nM T27812 D0X3CF 442879 IC50 = 175000 nM T27812 D0X8GC 45487773 IC50 = 10 nM T27812 D0X8LG 11243002 Ki = 33.1 nM T27812 D0XF5P 44592119 IC50 = 20 nM T27812 D0XY9E 3029724 IC50 > 100 nM T27812 D0Y1MJ 16102749 IC50 = 1900 nM T27812 D0Y3BI 11572135 IC50 = 24 nM T27812 D0Y5CG 45483467 Ki = 17 nM T27812 D0Y6GQ 44414862 IC50 = 230 nM T27812 D0Y7CS 44543118 IC50 > 100 nM T27812 D0Y7UJ 44592243 IC50 = 88 nM T27812 D0Y8UC 3929516 Ki = 3260 nM T27812 D0YZ3E 44435200 Ki = 3800 nM T27812 D0Z4UF 10524711 Ki = 2670 nM T27812 D0Z5GR 46230818 Ki > 4710 nM T27812 D0Z6YA 11289879 IC50 = 13 nM T27812 D0Z9OX 44414719 IC50 = 5.4 nM T27812 D0ZC3Q 44230732 Ki = 6 nM T27812 D0ZE4C 45141608 IC50 = 6900 nM T27812 D0ZU5W 22615724 Ki = 1140 nM T64969 D01PZD 5329098 IC50 > 100000 nM T64969 D03MNN 11341869 IC50 = 230 nM T64969 D03ZBT 11626560 IC50 = 681 nM T64969 D04LVK 57379345 IC50 = 28 nM T64969 D05NUH 54758501 IC50 = 10 nM T64969 D05UFG 10184653 IC50 = 0.19 nM T64969 D06IAR 60961 IC50 = 195000 nM T64969 D06XXH 11511120 IC50 = 1.8 nM T64969 D07POC 176870 Ki = 0.1 nM T64969 D08CDI 208908 Ki = 3 nM T64969 D08HVR 6047 IC50 = 900000 nM T64969 D08PIE 68165256 IC50 = 1 nM T64969 D09KTS 24821094 IC50 = 0.75 nM T64969 D09PQZ 71226662 IC50 > 2000 nM T64969 D09XZB 123631 IC50 = 0.1 nM T64969 D0AZ3C 5291 IC50 > 100000 nM T64969 D0B0AX 5328127 IC50 = 50000 nM T64969 D0C4RB 36314 IC50 > 10000 nM T64969 D0E6XR 3062316 IC50 = 180 nM T64969 D0EG1I 9926791 IC50 > 10000 nM T64969 D0G6QF 3081361 IC50 = 200 nM T64969 D0GY5Z 2244 IC50 > 10000 nM T64969 D0H0EQ 24826799 IC50 > 1000 nM T64969 D0IQ6P 25102847 IC50 = 19 nM T64969 D0J9ZR 4477 IC50 = 10500 nM T64969 D0K8KX 5280343 IC50 = 900 nM T64969 D0O8GK 71496458 IC50 = 0.421 nM T64969 D0OB0F 5328940 IC50 = 53 nM T64969 D0R0MW 5329102 IC50 = 140 nM T64969 D0R1QE 3672 IC50 > 10000 nM T64969 D0R1RS 3715 IC50 > 10000 nM T64969 D0W5HK 216239 IC50 = 43.5 nM T64969 D0W9WF 3825 IC50 > 10000 nM T64969 D0Y9EW 42611257 IC50 > 10000 nM T64969 D0Z5IU 1548887 IC50 > 10000 nM T64969 D00NYJ 42642648 IC50 = 7 nM T64969 D00RMC 6918508 IC50 = 3 nM T64969 D00YER 25127713 IC50 = 0.218 nM T64969 D01GFX 11640390 IC50 > 12500 nM T64969 D02BYZ 71667668 IC50 = 8 nM T64969 D02RJY 11442891 IC50 > 10000 nM T64969 D02TUL 118115473 IC50 > 50000 nM T64969 D02UFQ 11620908 IC50 = 1 nM T64969 D03LWG 53235510 IC50 > 10000 nM T64969 D04BFC 59174488 IC50 = 442 nM T64969 D06WRF 10458325 IC50 = 0.3 nM T64969 D07EHV 44814409 IC50 > 10000 nM T64969 D07HPJ 11476171 IC50 = 5200 nM T64969 D09TAB 25151352 IC50 > 10000 nM T64969 D0A1AQ 5329099 IC50 > 100000 nM T64969 D0BM7M 11488320 IC50 = 4 nM T64969 D0CN9Q 9874913 IC50 = 6400 nM T64969 D0D1GF 42642645 IC50 = 2990 nM T64969 D0E3TC 44259 IC50 = 0.38 nM T64969 D0G2QH 10297043 IC50 = 2 nM T64969 D0G5XV 135565884 IC50 = 2.6 nM T64969 D0HS5V 11234052 IC50 > 1900 nM T64969 D0I1DW 9808998 IC50 > 200000 nM T64969 D0K7FY 72703790 IC50 = 160.6 nM T64969 D0L4FS 5280961 IC50 = 0.1 ug.mL-1 T64969 D0LF1U 5287969 IC50 = 7600 nM T64969 D0M0XB 10302451 IC50 = 66 nM T64969 D0M4AV 57335384 IC50 = 1.6 nM T64969 D0O0LS 25141092 IC50 > 10000 nM T64969 D0O6WV 24794418 IC50 > 12500 nM T64969 D0P1CV 46191454 IC50 > 10000 nM T64969 D0P6DJ 151194 IC50 = 457.7 nM T64969 D0Q7RE 16007391 Ki > 10000 nM T64969 D0Q9CY 9915743 IC50 = 0.08 nM T64969 D0Q9UX 16718576 IC50 = 3069 nM T64969 D0QX8X 71479709 IC50 = 5800 nM T64969 D0R0LB 91668194 IC50 = 12 nM T64969 D0S3PO 6445562 IC50 = 8.02 nM T64969 D0S5RC 3025986 IC50 > 25000 nM T64969 D0U4FF 10437018 IC50 = 32 nM T64969 D0VF6E 1401 IC50 > 50000 nM T64969 D0X4MN 11597537 IC50 = 380 nM T64969 D0YB3W 156414 Ki = 0.11 nM T64969 D0Z4RC 24756910 IC50 = 2.4 nM T64969 D0ZN1R 68245 IC50 = 6.27 nM T64969 D03BNU 59604787 IC50 > 3500 nM T64969 D0LF0O 135441202 IC50 = 21000 nM T64969 D04SWX 56924694 IC50 = 113 nM T64969 D0NH9P 135 IC50 = 10 ug.mL-1 T64969 D0OE4F 4369496 IC50 > 100000 nM T64969 D00BPA 4592 IC50 = 440000 nM T64969 D01EFO 9864718 IC50 = 65000 nM T64969 D02YAQ 6603857 IC50 = 1 nM T64969 D03QTP 1697 Ki = 160 nM T64969 D03WTT 5468216 IC50 = 700 nM T64969 D04FHB 6918852 Ki > 5000 nM T64969 D07GFF 6918403 IC50 = 3.7 nM T64969 D08DBE 10344820 Ki = 35 nM T64969 D0A9KI 9863367 IC50 > 10 nM T64969 D0B3CT 9928668 IC50 = 29000 nM T64969 D0D5CJ 9818362 IC50 > 100000 nM T64969 D0F8DL 176155 IC50 > 33000 nM T64969 D0GZ7B 5328779 IC50 = 501.19 nM T64969 D0H8KG 5311382 IC50 = 44000 nM T64969 D0HO1S 6711154 IC50 = 700 nM T64969 D0IT6Q 3038522 IC50 > 30000 nM T64969 D0L5YF 5329032 IC50 = 50 nM T64969 D0Q7HO 4705 Ki = 0.006 nM T64969 D0T3ME 156422 IC50 = 3800 nM T64969 C0U5TZ 1302 IC50 > 10000 nM T64969 CB1VW3 1400 Ki = 199.53 nM T64969 C03TMS 1714 IC50 = 126.7 nM T64969 CO8C3E 2046 Ki = 150000 nM T64969 CH21PG 2428 IC50 = 0.008 nM T64969 C8HN2C 3798 IC50 = 29 nM T64969 C1BE5N 3799 IC50 = 10000 nM T64969 C2LS4F 3895 IC50 = 0.5 ug.mL-1 T64969 C0W4UD 3896 IC50 = 30 nM T64969 C2DUS8 4706 IC50 = 0.69 nM T64969 CBPM40 4878 IC50 = 480 nM T64969 CKZH57 5613 IC50 = 6500000 nM T64969 C2I3WC 5614 Ki = 155000 nM T64969 CQAO39 9210 IC50 = 27 nM T64969 CO7NY6 18091 Ki = 117000 nM T64969 C8K2FU 18606 IC50 > 1250000 nM T64969 CN31AP 19424 Ki = 67000 nM T64969 C12BXO 23905 IC50 = 225000 nM T64969 CL3H9Z 33296 IC50 > 325000 nM T64969 C0TMU5 37583 IC50 = 1400000 nM T64969 C4D5OH 44390 IC50 = 250000 nM T64969 C43WLX 57591 Ki = 50000 nM T64969 C62EPW 58857 Ki = 55000 nM T64969 CQD56Z 73299 IC50 > 20000 nM T64969 C63WLY 89644 IC50 = 6 ug.mL-1 T64969 CE4K5D 92516 IC50 > 50000 nM T64969 CI27WO 92970 Ki = 160000 nM T64969 C5JE2Z 104860 IC50 = 3.5 ug.mL-1 T64969 CF5B3H 121059 IC50 = 600000 nM T64969 C91ERH 128872 IC50 = 23 nM T64969 C6Y9CV 151193 IC50 > 10000 nM T64969 CRFU83 156413 IC50 = 1.5 nM T64969 CA5CO8 157820 IC50 > 100000 nM T64969 CI1NA5 159926 IC50 = 2.7 ug.mL-1 T64969 CI80NA 160436 IC50 > 50000 nM T64969 CV7W4J 176406 IC50 = 2511.89 nM T64969 C2P8XO 176871 IC50 = 70 nM T64969 CYBA43 177458 IC50 = 4 ug.mL-1 T64969 CPI83T 198909 IC50 = 4100 nM T64969 CRP4A8 244537 IC50 > 250000 nM T64969 C8MUX3 252473 Ki = 123000 nM T64969 C4C7HJ 282723 Ki > 400000 nM T64969 C61DPM 321779 Ki > 250000 nM T64969 CPF26C 324081 IC50 = 344 nM T64969 C9WA8F 341040 IC50 = 5600 nM T64969 CL1M8I 350716 IC50 > 50000 nM T64969 CV3XI1 354479 IC50 = 350 nM T64969 CZ5B0Y 367524 Ki > 400000 nM T64969 C0DI9H 375472 IC50 = 5000 nM T64969 C0M4OG 375473 IC50 = 3300 nM T64969 CMH0V9 382059 IC50 = 10 nM T64969 CQX5W6 390508 IC50 = 10000 nM T64969 CPF67R 402810 IC50 = 41900 nM T64969 CNP3M1 403661 IC50 = 320000 nM T64969 CC2R6G 409975 IC50 = 1800 nM T64969 CK0L4O 442514 IC50 = 3400 nM T64969 C4MNG8 445840 IC50 > 20000 nM T64969 C1YNB7 447721 IC50 > 10000 nM T64969 C1ZG2U 449087 IC50 > 10000 nM T64969 CT5O9L 519420 IC50 = 1500000 nM T64969 CSA52V 542795 IC50 > 20000 nM T64969 CVQ2Y4 589288 IC50 = 0.79 nM T64969 CO0U5E 616443 IC50 > 20000 nM T64969 C53PTU 616573 IC50 = 320 nM T64969 C2U6LB 643159 IC50 = 850000 nM T64969 C75EDQ 644355 IC50 > 30000 nM T64969 C5HPF3 644356 IC50 > 30000 nM T64969 CSA18D 651672 IC50 = 577 nM T64969 CJ0YU6 659954 IC50 = 912.01 nM T64969 CR3N8A 667645 Ki = 2200 nM T64969 CP91NX 677915 IC50 = 14590 nM T64969 CLEU84 689033 IC50 > 100000 nM T64969 CDE9V2 689424 IC50 = 19690 nM T64969 C5O0TJ 690158 IC50 = 23160 nM T64969 C7TPR6 690965 IC50 = 9050 nM T64969 C3Q6IY 694087 IC50 > 100000 nM T64969 C3V5KD 694921 IC50 > 250000 nM T64969 CX17CH 701322 IC50 = 63 nM T64969 C34EXB 702486 IC50 = 13930 nM T64969 CYO86G 703960 IC50 > 100000 nM T64969 C4BX6T 707914 IC50 = 560000 nM T64969 CD69IF 710163 IC50 > 625000 nM T64969 C65SGT 712193 IC50 = 842 nM T64969 C6D4HT 720879 IC50 = 325000 nM T64969 C6CJY8 725409 IC50 = 30 nM T64969 CTO15S 727131 IC50 = 10020 nM T64969 C9D7UY 727518 IC50 > 100000 nM T64969 C2CL6X 732134 IC50 = 5160 nM T64969 CKO38Q 732136 IC50 = 10230 nM T64969 C6AKG9 735124 IC50 = 56 nM T64969 C17UDE 735126 IC50 = 80 nM T64969 C4V7OW 736236 IC50 = 833000 nM T64969 CT7E1K 746495 Ki = 300000 nM T64969 C6ECP2 755464 IC50 = 11690 nM T64969 CWZY50 764334 IC50 = 15740 nM T64969 CPKI76 765318 IC50 = 9860 nM T64969 CXME85 766168 IC50 = 13710 nM T64969 CB30XT 778859 IC50 = 16170 nM T64969 CQB03J 780790 IC50 = 12290 nM T64969 C7EHR1 787183 IC50 = 12690 nM T64969 CLU06E 792233 IC50 = 14580 nM T64969 C73TME 811665 IC50 = 12320 nM T64969 CTX13N 814517 IC50 = 460 nM T64969 CB27WS 849733 IC50 > 10000 nM T64969 CW56XG 875024 IC50 = 7370 nM T64969 CP40SX 889945 IC50 = 5720 nM T64969 C5GMN8 935994 IC50 = 149 nM T64969 CXB5A2 964113 IC50 > 100000 nM T64969 CW7FM4 967629 IC50 = 26060 nM T64969 C7SD1U 1007600 IC50 = 3500 nM T64969 C9DBI2 1011523 IC50 = 9700 nM T64969 C0NF2R 1018252 IC50 = 5600 nM T64969 CR8F6B 1035343 IC50 > 100000 nM T64969 CEF7B3 1086535 IC50 = 8400 nM T64969 C9U7NK 1128774 IC50 = 76700 nM T64969 CQWX85 1304420 IC50 = 15000 nM T64969 CJP04L 1474852 IC50 = 0.07244 nM T64969 CYQ90E 1474874 IC50 > 1000 nM T64969 C6OC3G 1474877 IC50 = 10 nM T64969 CC3A8B 1474883 IC50 = 3.8 nM T64969 CK3QN1 1475063 IC50 = 19.1 nM T64969 C3SGW1 1490236 IC50 = 3000 nM T64969 CMYK57 1500232 IC50 = 24830 nM T64969 C84MXV 1500233 IC50 > 30000 nM T64969 CDB17F 1538822 IC50 = 18500 nM T64969 CG73KY 1550166 Ki = 1400000 nM T64969 C2BCN0 1550170 IC50 = 833000 nM T64969 CRQ82G 1558661 Ki = 1350000 nM T64969 CSA69X 1637668 IC50 = 9350 nM T64969 C6ZY1V 1641261 IC50 > 20000 nM T64969 C5WM1Q 1723871 IC50 = 8600 nM T64969 CL6IN7 1742852 IC50 = 74300 nM T64969 CVA45M 1810492 IC50 = 23100 nM T64969 C1P4FC 1838043 IC50 = 12022.64 nM T64969 CDC7Q4 1900460 IC50 = 35800 nM T64969 C71YPT 2103474 IC50 = 35 nM T64969 CZ2B4M 2358462 IC50 > 100000 nM T64969 CXA1L7 2365265 IC50 > 100000 nM T64969 CEF62M 2379240 IC50 > 100000 nM T64969 CS6RH2 2385464 IC50 = 5888.44 nM T64969 C7EB0A 2385467 IC50 = 2000 nM T64969 CKT64G 2396126 IC50 > 10000 nM T64969 C6T0OJ 2400783 IC50 = 2980 nM T64969 CKE7P2 2725645 IC50 = 200 nM T64969 C31KAP 2743369 IC50 = 54 nM T64969 C5ON0G 2744121 IC50 > 100000 nM T64969 C9IWU0 2789324 IC50 = 50 nM T64969 C4POJ7 2795373 IC50 = 260000 nM T64969 CG43CZ 2802451 IC50 = 2520 nM T64969 C8S0UP 2806990 IC50 = 45500 nM T64969 CV7Y5T 2807058 IC50 = 1500 nM T64969 C8VD6N 2808930 IC50 > 3240 nM T64969 C0KB3P 2810857 IC50 = 11100 nM T64969 CEX1W9 2811342 IC50 > 100000 nM T64969 CSA5I6 2839887 IC50 = 6270 nM T64969 C9VUX8 2843335 IC50 = 16630 nM T64969 C3BJP7 2943601 IC50 > 10000 nM T64969 C8HAL7 2983225 IC50 = 38430 nM T64969 CFVK40 3008950 IC50 > 50000 nM T64969 CD8UW1 3008956 IC50 = 200 nM T64969 CCD93P 3008957 IC50 = 1240 nM T64969 CU64VM 3008958 IC50 = 1670 nM T64969 C8F0KM 3008959 IC50 = 4310 nM T64969 CV8R9Z 3008960 IC50 = 6160 nM T64969 C8EZ6O 3008961 IC50 = 9190 nM T64969 CX95SU 3008962 IC50 = 12620 nM T64969 C9B2MN 3008963 IC50 = 17420 nM T64969 C9E7BW 3008964 IC50 = 19770 nM T64969 CGK91Q 3008965 IC50 > 50000 nM T64969 CHGP54 3035187 IC50 = 0.8 nM T64969 CJBX04 3039851 IC50 = 1500 nM T64969 CHK3W2 3135836 IC50 = 92400 nM T64969 C2SM4G 3138425 IC50 = 81600 nM T64969 CCN9D5 3142817 IC50 = 280 nM T64969 CUK5Y1 3374314 IC50 = 20000 nM T64969 CW74LV 3564138 IC50 > 10000 nM T64969 C3QSK2 3677514 IC50 = 72400 nM T64969 C46IJS 3724145 IC50 = 5110 nM T64969 CCUW85 4205046 IC50 = 4300 nM T64969 CPHI06 4321095 IC50 > 100000 nM T64969 CZB15R 4350438 IC50 = 2000 nM T64969 CM5VN6 4600415 IC50 = 88670 nM T64969 C8O9MN 4616059 IC50 = 1330 nM T64969 C2W4OD 4677622 IC50 = 20190 nM T64969 CN7MT6 4750207 IC50 = 31000 nM T64969 CB3G6R 4913175 IC50 = 200 nM T64969 CSI43N 5083839 IC50 = 28690 nM T64969 C1BPI8 5280569 IC50 = 7670 nM T64969 C8N6AY 5281377 IC50 > 100 ug.mL-1 T64969 C4JB3P 5281801 IC50 = 3 ug.mL-1 T64969 C0FLB1 5281811 IC50 = 3300 nM T64969 CTID76 5282335 IC50 > 25000 nM T64969 CY28LS 5293755 IC50 > 100000 nM T64969 CW26CH 5311106 IC50 > 20000 nM T64969 C4VTS3 5327723 IC50 > 100000 nM T64969 C6UL3A 5327821 IC50 = 220 nM T64969 CR3OF4 5327822 IC50 = 160 nM T64969 C9QMX2 5327823 IC50 = 58 nM T64969 CA4G1B 5327824 IC50 = 84 nM T64969 CY2NC3 5327825 IC50 = 250 nM T64969 CDT07K 5327826 IC50 < 800 nM T64969 CG36XB 5327827 IC50 = 130 nM T64969 CF3Y6G 5327828 IC50 = 30 nM T64969 CY1Z9E 5327829 IC50 = 8 nM T64969 CI51CH 5327830 IC50 = 8 nM T64969 CUAW78 5327831 IC50 = 4 nM T64969 CC9US2 5327832 IC50 > 100000 nM T64969 CVGK98 5327833 IC50 = 5 nM T64969 CGWP86 5327834 IC50 = 29 nM T64969 C10RVD 5327835 IC50 = 3 nM T64969 CD6B2A 5327836 IC50 = 26 nM T64969 CY1O6K 5327837 IC50 = 8 nM T64969 C1K8CJ 5327838 IC50 = 7 nM T64969 CP15JO 5327839 IC50 = 19 nM T64969 CWT9S8 5327840 IC50 = 26 nM T64969 C5EWD2 5327841 IC50 = 96 nM T64969 C67JVQ 5327843 IC50 = 270 nM T64969 CY23QP 5327844 IC50 = 5 nM T64969 CN1X4Z 5327845 IC50 = 270 nM T64969 C6TGI1 5327846 IC50 = 2 nM T64969 CEMR07 5327847 IC50 = 24200 nM T64969 CB90GI 5327848 IC50 = 1500 nM T64969 CMC76E 5327864 IC50 = 5600 nM T64969 C43JFT 5327866 IC50 > 50000 nM T64969 C4ZW0Q 5327868 IC50 = 7500 nM T64969 CY82TU 5327869 IC50 = 4500 nM T64969 CL4OG5 5327870 IC50 > 5000 nM T64969 CYGA64 5327871 IC50 = 4400 nM T64969 CZE87D 5327872 IC50 > 50000 nM T64969 C7XOK5 5327873 IC50 > 5000 nM T64969 CQK5Z0 5327874 IC50 > 50000 nM T64969 CS0Q4N 5327875 IC50 > 50000 nM T64969 CI96EG 5327876 IC50 = 1400 nM T64969 CT86OE 5327877 IC50 > 5000 nM T64969 C23EZX 5327878 IC50 = 8700 nM T64969 C63SAG 5327879 IC50 = 210 nM T64969 CT94BD 5327880 IC50 = 4500 nM T64969 CNRS28 5327881 IC50 > 5000 nM T64969 CD43FT 5327882 IC50 > 5000 nM T64969 CX39AM 5327883 IC50 > 5000 nM T64969 CZWG61 5327884 IC50 = 1000 nM T64969 C3P8CG 5327885 IC50 = 260 nM T64969 CWZ8H3 5327886 IC50 = 200 nM T64969 CC7VR3 5327887 IC50 = 510 nM T64969 CG7Q3R 5327888 IC50 = 1300 nM T64969 CYRW80 5327889 IC50 = 910 nM T64969 C7W8IJ 5327890 IC50 = 490 nM T64969 CJ28SO 5327891 IC50 > 5000 nM T64969 C82PDN 5327892 IC50 = 670 nM T64969 C52MYD 5327893 IC50 = 480 nM T64969 C4ET5H 5327894 IC50 = 66 nM T64969 CJ5VO8 5327895 IC50 = 30 nM T64969 CDA78E 5327896 IC50 = 220 nM T64969 CQ0ZP3 5327897 IC50 = 150 nM T64969 COQH79 5327899 IC50 = 250 nM T64969 C9R8DP 5327900 IC50 = 330 nM T64969 CVB9L3 5327902 IC50 > 50000 nM T64969 C7EK0Z 5327903 IC50 = 700 nM T64969 CN71AK 5327916 IC50 = 190 nM T64969 C5JI1A 5327917 IC50 = 220 nM T64969 C4CWI1 5327918 IC50 = 80 nM T64969 CQ0J3U 5328014 IC50 = 7000 nM T64969 C0FCR1 5328015 IC50 = 10000 nM T64969 C5VW6K 5328016 IC50 > 50000 nM T64969 C5IL6F 5328017 IC50 > 1000 nM T64969 C6RHB3 5328018 IC50 = 756 nM T64969 C5FXG1 5328019 IC50 = 5500 nM T64969 CPF5M1 5328020 IC50 > 10000 nM T64969 CKOI31 5328021 IC50 > 100000 nM T64969 CV5IX3 5328022 IC50 > 100000 nM T64969 CK31WA 5328023 IC50 > 1000 nM T64969 CFH4N1 5328024 IC50 = 8000 nM T64969 C89PLV 5328025 IC50 > 10000 nM T64969 CWE6K5 5328026 IC50 = 4900 nM T64969 CH5R7E 5328027 IC50 > 10000 nM T64969 CU6F0M 5328028 IC50 = 508 nM T64969 C0N4ZK 5328029 IC50 = 200 nM T64969 CYVQ61 5328030 IC50 = 5900 nM T64969 CP4AW6 5328031 IC50 > 1000 nM T64969 CH0J3D 5328032 IC50 = 58 nM T64969 C6R2HK 5328033 IC50 > 10000 nM T64969 CG2PT3 5328034 IC50 > 10000 nM T64969 C8BEX5 5328035 IC50 > 10000 nM T64969 C7KO4J 5328037 IC50 = 56 nM T64969 C7NAH0 5328039 IC50 = 439 nM T64969 CIRD30 5328040 IC50 = 139 nM T64969 CCL34N 5328041 IC50 = 897 nM T64969 C0SF3M 5328043 IC50 = 30 nM T64969 C8N1PH 5328044 IC50 = 1000 nM T64969 CCZP83 5328046 IC50 = 10 nM T64969 CG94OR 5328047 IC50 > 10000 nM T64969 C1AEK5 5328048 IC50 = 105 nM T64969 C0W1KQ 5328049 IC50 = 974 nM T64969 C5VS7Z 5328051 IC50 = 250 nM T64969 C8MK4H 5328052 IC50 = 1250 nM T64969 C5EO6F 5328053 IC50 = 40 nM T64969 C3NP1J 5328054 IC50 = 65000 nM T64969 CFS1Q9 5328055 IC50 = 240 nM T64969 C5MB0W 5328056 IC50 = 90 nM T64969 C5U7TE 5328057 IC50 = 10000 nM T64969 CLG58H 5328058 IC50 = 15 nM T64969 CK3W0S 5328059 IC50 = 4700 nM T64969 CECV59 5328060 IC50 = 3710 nM T64969 C6QT8H 5328061 IC50 = 130 nM T64969 CL2KB9 5328062 IC50 = 670 nM T64969 CT87KZ 5328063 IC50 = 5250 nM T64969 CFSQ97 5328064 IC50 = 1550 nM T64969 CIWL47 5328065 IC50 = 5900 nM T64969 C4AY9I 5328066 IC50 = 69000 nM T64969 CN7I4H 5328067 IC50 = 1790 nM T64969 CA02CD 5328068 IC50 = 4860 nM T64969 C6MZ2K 5328069 IC50 = 840 nM T64969 C4CGO6 5328070 IC50 = 120 nM T64969 C68BQO 5328071 IC50 = 260 nM T64969 CEJB59 5328072 IC50 = 70 nM T64969 C1B7ZI 5328073 IC50 = 40 nM T64969 C0VL9E 5328074 IC50 > 10000 nM T64969 CW73VX 5328075 IC50 > 10000 nM T64969 CJ6CB8 5328076 IC50 > 10000 nM T64969 CJ6PO5 5328078 IC50 = 4250 nM T64969 C1N8WQ 5328079 IC50 = 10100 nM T64969 C58USW 5328080 IC50 > 10000 nM T64969 C5I8CA 5328081 IC50 = 1670 nM T64969 CM5EX7 5328082 IC50 = 1000 nM T64969 C1U0NE 5328083 IC50 = 2460 nM T64969 CRA1U0 5328084 IC50 = 10000 nM T64969 C1BC5V 5328085 IC50 = 1950 nM T64969 C5NKF7 5328086 IC50 = 8000 nM T64969 C6ID3P 5328087 IC50 = 100000 nM T64969 C6XJ8Q 5328088 IC50 = 2870 nM T64969 C7SC8N 5328089 IC50 > 100000 nM T64969 C94MXF 5328090 IC50 = 230 nM T64969 C8FI2S 5328091 IC50 > 10000 nM T64969 C0M5QH 5328092 IC50 > 10000 nM T64969 C05WQF 5328093 IC50 > 100000 nM T64969 CEB5H2 5328094 IC50 = 10000 nM T64969 C0XFQ1 5328095 IC50 > 100000 nM T64969 CCZ96X 5328096 IC50 = 1800 nM T64969 CW4XA5 5328097 IC50 = 3300 nM T64969 CHS5A1 5328098 IC50 > 100000 nM T64969 C4IJ7Z 5328099 IC50 = 3500 nM T64969 C4G6XV 5328100 Ki = 3100 nM T64969 CMTP83 5328101 IC50 = 4700 nM T64969 CH4P3L 5328102 IC50 = 13000 nM T64969 C5R9ZI 5328103 IC50 = 4600 nM T64969 CM06LQ 5328104 IC50 = 6900 nM T64969 CPT61U 5328112 IC50 = 450 nM T64969 CXR9K1 5328115 IC50 = 6200 nM T64969 CM0H5O 5328117 IC50 = 610 nM T64969 CDM98R 5328125 IC50 = 6680 nM T64969 CDY2O3 5328134 IC50 = 1300 nM T64969 CC1O0M 5328135 IC50 = 240 nM T64969 C14LVT 5328137 IC50 = 1000 nM T64969 COT45A 5328149 IC50 = 150 nM T64969 CF3AM9 5328157 IC50 = 980 nM T64969 CT9SO8 5328158 IC50 = 880 nM T64969 CJA36I 5328171 IC50 = 720 nM T64969 C5CZF2 5328186 IC50 = 55 nM T64969 CVF39K 5328187 IC50 = 770 nM T64969 C8SQG9 5328188 IC50 = 575.44 nM T64969 C2L4GQ 5328189 IC50 = 5000 nM T64969 C5L7OH 5328190 IC50 = 120 nM T64969 C6G8MS 5328191 IC50 = 100 nM T64969 CR6UC1 5328192 IC50 = 2 nM T64969 CSE29Z 5328193 IC50 = 0.25 nM T64969 CE2X5M 5328194 IC50 = 0.35 nM T64969 CDN5A9 5328195 IC50 = 3.3 nM T64969 CE3OP6 5328196 IC50 = 12000 nM T64969 CAU43H 5328197 IC50 = 6100 nM T64969 CR5Q3J 5328198 IC50 = 810 nM T64969 C9B8MI 5328199 IC50 = 540 nM T64969 C0V3QG 5328200 IC50 > 10000 nM T64969 C48GSA 5328201 IC50 = 0.89 nM T64969 C2TVO1 5328202 IC50 = 0.24 nM T64969 CQ3SK4 5328203 IC50 = 4 nM T64969 C3DXQ1 5328204 IC50 = 84 nM T64969 CL3X6O 5328205 IC50 = 12.02 nM T64969 CMQ0D5 5328207 IC50 = 40 nM T64969 C8VF0X 5328208 IC50 = 4 nM T64969 CASZ78 5328209 IC50 = 12 nM T64969 CCQX42 5328210 IC50 = 11 nM T64969 CEK4W5 5328211 IC50 = 162.18 nM T64969 CH89ZL 5328212 IC50 = 3.802 nM T64969 CB35RO 5328213 IC50 = 6.5 nM T64969 CX7CS9 5328214 IC50 = 53 nM T64969 CXWA71 5328215 IC50 = 68 nM T64969 CX4FR7 5328216 IC50 = 2000 nM T64969 CA6M1B 5328217 IC50 = 28 nM T64969 C1SR4I 5328218 IC50 = 15 nM T64969 CQ3MT4 5328219 IC50 = 25.12 nM T64969 C5W4EO 5328220 IC50 = 15 nM T64969 CPBJ63 5328221 IC50 = 0.1738 nM T64969 CA0E1F 5328222 IC50 = 105 nM T64969 CE9H1T 5328223 IC50 = 1370 nM T64969 CA4C8N 5328224 IC50 > 10000 nM T64969 CIEL17 5328225 IC50 > 10000 nM T64969 CCX4R2 5328226 IC50 = 463 nM T64969 CKY7Z5 5328227 IC50 = 152 nM T64969 CO12GB 5328228 IC50 = 0.67 nM T64969 CTV8F0 5328229 IC50 > 10000 nM T64969 CZG75R 5328230 IC50 = 128 nM T64969 COH17Q 5328231 IC50 = 0.072 nM T64969 CYU3Z1 5328232 IC50 = 113 nM T64969 CD8JS2 5328233 IC50 = 0.29 nM T64969 C5FY4G 5328234 IC50 = 0.01 nM T64969 C5GCU1 5328235 IC50 = 1.32 nM T64969 CJN72V 5328236 IC50 = 22 nM T64969 CV7UC8 5328237 IC50 = 203 nM T64969 CZE57H 5328238 IC50 = 29 nM T64969 C3TNY6 5328239 IC50 = 272 nM T64969 C5LS7N 5328240 IC50 = 44 nM T64969 C4S0YJ 5328241 IC50 = 0.34 nM T64969 CP4Y5S 5328242 IC50 = 0.44 nM T64969 C3EF7M 5328243 IC50 = 0.39 nM T64969 CAE24W 5328246 IC50 = 1.7 nM T64969 CH62XU 5328247 IC50 = 1460 nM T64969 C7XLU4 5328248 IC50 = 100 nM T64969 CS60WL 5328249 IC50 = 35.48 nM T64969 C6CU9X 5328250 IC50 = 29 nM T64969 CRW56D 5328251 IC50 = 13 nM T64969 CHZ78I 5328252 IC50 = 16 nM T64969 C1LX5E 5328253 IC50 = 14 nM T64969 C3EB6U 5328254 IC50 = 39 nM T64969 CUAH85 5328256 IC50 = 2030 nM T64969 CWCJ02 5328257 IC50 = 51 nM T64969 CC0F5Z 5328258 IC50 = 0.13 nM T64969 CY0AH6 5328259 IC50 = 40 nM T64969 C8UG0Z 5328260 IC50 = 124 nM T64969 CVK13Z 5328261 IC50 = 0.006 nM T64969 CVT30D 5328262 IC50 = 2.63 nM T64969 C4ML9Z 5328263 IC50 = 2.3 nM T64969 CZU8N4 5328264 IC50 = 9 nM T64969 CJU52L 5328265 IC50 > 10 nM T64969 C7QH8D 5328266 IC50 = 688 nM T64969 C5C4BE 5328267 IC50 = 954.99 nM T64969 CCN5Y6 5328268 IC50 = 684 nM T64969 CE1Q2B 5328269 IC50 = 52 nM T64969 CA4R3X 5328270 IC50 = 331.13 nM T64969 C8BP2W 5328271 IC50 = 263 nM T64969 C5YRH9 5328272 IC50 = 603 nM T64969 C5O7VR 5328273 IC50 = 34 nM T64969 CE3JU1 5328274 IC50 = 53 nM T64969 C7WD6E 5328275 IC50 = 18 nM T64969 C1ORZ0 5328276 IC50 = 44 nM T64969 C2L3RB 5328277 IC50 = 3.1 nM T64969 CD20TF 5328278 IC50 = 9.6 nM T64969 CQO15H 5328279 IC50 = 4.3 nM T64969 CNEF93 5328280 IC50 = 0.37 nM T64969 CR2W7Q 5328281 IC50 = 12 nM T64969 CA2CP7 5328282 IC50 = 39.81 nM T64969 CS16CZ 5328283 IC50 = 3.7 nM T64969 CEF8A6 5328284 IC50 = 52.48 nM T64969 CUFW39 5328285 IC50 = 21.88 nM T64969 C1PC0U 5328286 IC50 = 1.6 nM T64969 CI7H3A 5328287 IC50 = 41 nM T64969 C8O2FY 5328288 IC50 = 21 nM T64969 CQ1OD4 5328289 IC50 = 3.7 nM T64969 C0W1HD 5328290 IC50 = 77.62 nM T64969 C0R1WK 5328291 IC50 = 5.1 nM T64969 C0QUZ5 5328292 IC50 = 135 nM T64969 CTI8W5 5328293 IC50 = 9.7 nM T64969 C8THM7 5328294 IC50 = 4.8 nM T64969 CJY1D0 5328295 IC50 = 81 nM T64969 C7FQ0J 5328296 IC50 = 3.388 nM T64969 CI32AD 5328297 IC50 = 0.72 nM T64969 C49IVK 5328298 IC50 = 0.24 nM T64969 C03MPD 5328299 IC50 = 2.57 nM T64969 CN7T3V 5328300 IC50 = 0.92 nM T64969 CL6HI8 5328301 IC50 = 3.2 nM T64969 C0JO8H 5328302 IC50 = 14 nM T64969 CVZQ92 5328303 IC50 = 12 nM T64969 CMV6R1 5328304 IC50 = 4.786 nM T64969 CSGC46 5328305 IC50 = 3.2 nM T64969 C0HIY2 5328306 IC50 = 44.67 nM T64969 C75QGA 5328307 IC50 = 8.71 nM T64969 CED9Z1 5328308 IC50 = 7.4 nM T64969 C5LC3J 5328309 IC50 = 8.318 nM T64969 C2RB9W 5328310 IC50 = 39.81 nM T64969 CT1V0S 5328311 IC50 = 3.236 nM T64969 CH1RI6 5328312 IC50 = 1.9 nM T64969 C82PRW 5328313 IC50 = 5.4 nM T64969 C5IN3X 5328314 IC50 = 0.74 nM T64969 CZ1VX5 5328315 IC50 = 4.898 nM T64969 CE6H9B 5328316 IC50 = 9.12 nM T64969 CH1ZV3 5328317 IC50 = 1.2 nM T64969 CEX9D0 5328318 IC50 = 7.1 nM T64969 CW4MH8 5328319 IC50 = 0.51 nM T64969 C2X4IR 5328320 IC50 = 0.91 nM T64969 C8CT3Z 5328321 IC50 = 1.5 nM T64969 C1UC9A 5328322 IC50 = 0.61 nM T64969 C4MO0D 5328323 IC50 = 0.2818 nM T64969 CLGB27 5328324 IC50 = 15.85 nM T64969 CY0AM6 5328325 IC50 = 1.4 nM T64969 CX7JZ8 5328326 IC50 = 1.413 nM T64969 C4CJW1 5328327 IC50 = 5.37 nM T64969 C80JRW 5328328 IC50 = 9.3 nM T64969 CWM81T 5328329 IC50 = 5.6 nM T64969 CZ8GQ5 5328330 IC50 = 3.5 nM T64969 C27YZX 5328331 IC50 = 7.2 nM T64969 C4BXI1 5328332 IC50 = 2550 nM T64969 CF8X6A 5328333 IC50 = 13 nM T64969 CHR91V 5328334 IC50 = 83.18 nM T64969 CZ1M2D 5328335 IC50 = 1.5 nM T64969 CSH09Q 5328336 IC50 = 0.76 nM T64969 C5S9YM 5328337 IC50 = 0.95 nM T64969 CFR57D 5328338 IC50 = 3.8 nM T64969 CUN2R4 5328339 IC50 = 35 nM T64969 C0NY7V 5328340 IC50 = 0.81 nM T64969 C0LDH1 5328341 IC50 = 2.9 nM T64969 CQ6ZM5 5328342 IC50 = 0.2512 nM T64969 CC2VT4 5328343 IC50 = 2.3 nM T64969 CUY75Z 5328344 IC50 = 380 nM T64969 CA6KZ4 5328345 IC50 = 17 nM T64969 CB3OP9 5328346 IC50 = 4.3 nM T64969 C1R7LX 5328347 IC50 = 4 nM T64969 CA1VR6 5328348 IC50 = 2.3 nM T64969 CK92CS 5328349 IC50 = 3 nM T64969 COI17R 5328350 IC50 = 0.19 nM T64969 C34OXD 5328351 IC50 = 0.22 nM T64969 CB4AJ3 5328352 IC50 = 0.18 nM T64969 C7ABZ1 5328353 IC50 = 0.56 nM T64969 CDV19S 5328354 IC50 = 1.1 nM T64969 CN62LQ 5328355 IC50 = 1.2 nM T64969 CIW27V 5328356 IC50 = 1.8 nM T64969 C1D0YT 5328357 IC50 = 4.6 nM T64969 C0X4VK 5328358 IC50 = 1.7 nM T64969 CV1L9N 5328359 IC50 = 8.1 nM T64969 CC4O6Y 5328360 IC50 = 0.65 nM T64969 CE3UW4 5328361 IC50 = 1 nM T64969 CU65HL 5328363 IC50 = 0.93 nM T64969 C7L1MN 5328364 IC50 = 230 nM T64969 C6S4LT 5328365 IC50 = 1.5 nM T64969 CG4RZ8 5328366 IC50 = 1.2 nM T64969 C6K4VL 5328367 IC50 = 0.78 nM T64969 CYLS53 5328368 IC50 = 1.7 nM T64969 CJY62E 5328369 IC50 = 102 nM T64969 C5EO4G 5328370 IC50 = 0.28 nM T64969 CP37XG 5328371 IC50 = 0.44 nM T64969 C0X8JK 5328372 IC50 = 449 nM T64969 C0EFY7 5328373 IC50 = 0.19 nM T64969 C7R3YC 5328374 IC50 = 1.1 nM T64969 C8IXG0 5328375 IC50 = 3.1 nM T64969 CE4R1Q 5328376 IC50 = 0.45 nM T64969 C0ON1H 5328377 IC50 = 2.8 nM T64969 CWPM74 5328378 IC50 = 1.5 nM T64969 C2QNS7 5328379 IC50 = 1.8 nM T64969 C3MHX9 5328380 IC50 = 1.3 nM T64969 CG0W7E 5328381 IC50 = 117 nM T64969 CJF0H4 5328382 IC50 = 1 nM T64969 CM96IG 5328383 IC50 = 11 nM T64969 C2REG3 5328387 IC50 = 419 nM T64969 CTBV20 5328388 IC50 = 50 nM T64969 CG3J4S 5328389 IC50 > 100000 nM T64969 CJY35F 5328391 IC50 = 264 nM T64969 C5FY3T 5328392 IC50 = 31 nM T64969 CXNL13 5328393 IC50 = 742 nM T64969 CF7J4M 5328394 IC50 = 4100 nM T64969 CF5SL0 5328396 IC50 = 147 nM T64969 CDEY49 5328397 IC50 = 1.2 nM T64969 C51IFH 5328398 IC50 = 4270 nM T64969 CEG9H2 5328399 IC50 = 191 nM T64969 C84GLZ 5328400 IC50 = 538 nM T64969 C6JA7G 5328401 IC50 = 1.8 nM T64969 CO17CE 5328407 IC50 = 2.1 nM T64969 CBO8C1 5328408 IC50 = 47 nM T64969 C61RXT 5328409 IC50 = 0.27 nM T64969 CVED61 5328412 IC50 = 42 nM T64969 CR6LU1 5328414 IC50 = 80 nM T64969 C1GL9F 5328416 IC50 = 19.8 nM T64969 CU2N1B 5328422 IC50 > 1000 nM T64969 CV2D5L 5328423 IC50 = 732 nM T64969 C46BDX 5328425 IC50 = 740 nM T64969 CJN93G 5328535 IC50 = 14900 nM T64969 CIV92Z 5328536 IC50 > 100000 nM T64969 CW8B1J 5328537 IC50 = 100000 nM T64969 CPN2E4 5328538 IC50 > 100000 nM T64969 CLQ9B1 5328539 IC50 = 1620 nM T64969 CA7LK0 5328540 IC50 = 6700 nM T64969 CW59PN 5328541 IC50 > 100000 nM T64969 CWB7K0 5328542 IC50 > 100000 nM T64969 C3UWT2 5328543 IC50 = 6700 nM T64969 C5FA3P 5328544 IC50 > 100000 nM T64969 C9DL4S 5328545 IC50 > 100000 nM T64969 C2PF4N 5328546 IC50 > 100000 nM T64969 C6UWZ8 5328547 IC50 > 100000 nM T64969 C9LMP7 5328548 IC50 > 100000 nM T64969 C3D5KN 5328549 IC50 > 100000 nM T64969 CL7JE8 5328550 IC50 = 10200 nM T64969 CV08ZJ 5328551 IC50 = 53000 nM T64969 CEQ5A8 5328552 IC50 = 14000 nM T64969 C0MP1C 5328553 IC50 = 18000 nM T64969 C3QA9X 5328554 IC50 = 33000 nM T64969 C6DN3V 5328555 IC50 > 100000 nM T64969 C6CMP2 5328556 IC50 = 9300 nM T64969 CQA3V1 5328557 IC50 = 35000 nM T64969 C3UAX9 5328558 IC50 = 4200 nM T64969 CS8A1P 5328559 IC50 = 3100 nM T64969 C3NC0W 5328560 IC50 = 21000 nM T64969 CXOP18 5328561 IC50 > 100000 nM T64969 C09UBN 5328562 IC50 = 8400 nM T64969 C71VUG 5328563 IC50 = 2900 nM T64969 COGL89 5328564 IC50 = 1500 nM T64969 CP5YX1 5328565 IC50 = 18000 nM T64969 C3WH4C 5328566 IC50 = 8300 nM T64969 C0QYJ7 5328567 IC50 > 100000 nM T64969 CHW4Q7 5328568 IC50 > 100000 nM T64969 CB9UI5 5328569 IC50 = 38000 nM T64969 CVEY01 5328570 IC50 = 32000 nM T64969 C3U1QJ 5328571 IC50 = 47000 nM T64969 CP5H9N 5328572 IC50 = 89000 nM T64969 C64XYH 5328573 IC50 = 16000 nM T64969 CBE9M4 5328574 IC50 = 9400 nM T64969 C5QE9H 5328575 IC50 = 68000 nM T64969 CE9PW4 5328576 IC50 = 12000 nM T64969 CJ78UZ 5328577 IC50 = 25000 nM T64969 C9S1MH 5328578 IC50 = 850 nM T64969 CE62YD 5328579 IC50 = 44000 nM T64969 C72KTF 5328580 IC50 = 7400 nM T64969 CG38AH 5328581 IC50 = 100000 nM T64969 C5HB9Z 5328582 IC50 = 8500 nM T64969 CGDE60 5328583 IC50 = 24000 nM T64969 COF98M 5328584 IC50 = 51000 nM T64969 C23LDB 5328585 IC50 > 100000 nM T64969 CXN72C 5328586 IC50 = 28000 nM T64969 CAT93L 5328587 IC50 = 14000 nM T64969 CA9PL4 5328588 IC50 = 100000 nM T64969 CQDX90 5328589 IC50 = 100000 nM T64969 CLZ2T7 5328590 IC50 = 22000 nM T64969 CMP24I 5328591 IC50 = 100000 nM T64969 C0TX2I 5328592 IC50 = 10000 nM T64969 C9JLN6 5328593 IC50 = 100000 nM T64969 C42LEK 5328594 IC50 > 100000 nM T64969 CVF12E 5328595 IC50 > 100000 nM T64969 CGN3C9 5328596 IC50 = 20000 nM T64969 C91NOL 5328597 IC50 > 100000 nM T64969 C0PB9W 5328598 IC50 = 4300 nM T64969 C9P3LY 5328599 IC50 = 11400 nM T64969 CQNB13 5328600 IC50 > 100000 nM T64969 CK7IA1 5328601 IC50 > 100000 nM T64969 CNI91T 5328602 IC50 = 5300 nM T64969 C3AW9S 5328603 IC50 = 40500 nM T64969 CWEA08 5328604 IC50 > 100000 nM T64969 CCM96I 5328605 IC50 = 54100 nM T64969 C9NVC5 5328606 IC50 = 5000 nM T64969 CDX4Z7 5328607 IC50 > 100000 nM T64969 CB1S3D 5328608 IC50 > 100000 nM T64969 C7WL3M 5328609 IC50 = 3600 nM T64969 C69QIE 5328610 IC50 > 100000 nM T64969 C09SPY 5328611 IC50 = 44000 nM T64969 CO2CR8 5328612 IC50 > 100000 nM T64969 CR3W8H 5328613 IC50 > 100000 nM T64969 CB2HD4 5328614 IC50 = 6500 nM T64969 C5GWD8 5328615 IC50 = 9900 nM T64969 C0MU7G 5328616 IC50 = 100000 nM T64969 CH1X6G 5328617 IC50 = 22300 nM T64969 CR02JQ 5328618 IC50 = 1000 nM T64969 CP8G4Z 5328619 IC50 > 100000 nM T64969 C8YS2H 5328620 IC50 > 100000 nM T64969 CM80FN 5328621 IC50 > 100000 nM T64969 C16JYR 5328622 IC50 > 100000 nM T64969 CL6QD5 5328623 IC50 > 100000 nM T64969 CFB26C 5328624 IC50 > 100000 nM T64969 C38PSR 5328744 IC50 > 250000 nM T64969 CJLU79 5328746 IC50 = 532000 nM T64969 CGM84A 5328747 IC50 = 800000 nM T64969 C71JTL 5328748 IC50 = 820000 nM T64969 CA9RY2 5328749 IC50 = 1480000 nM T64969 C2HDP0 5328750 IC50 = 1800000 nM T64969 C7LS0I 5328751 IC50 = 2200000 nM T64969 C6J4FI 5328752 IC50 > 2500000 nM T64969 CY9UG7 5328754 IC50 = 2500 nM T64969 CY8U9E 5328756 IC50 = 12500 nM T64969 CSZK53 5328757 IC50 = 26000 nM T64969 C46ZGF 5328758 IC50 = 60000 nM T64969 CX2G6U 5328759 IC50 = 1200000 nM T64969 CND59O 5328761 IC50 = 560 nM T64969 C68MGU 5328762 IC50 = 880 nM T64969 CN8L0R 5328764 IC50 = 1540 nM T64969 C2B0HF 5328765 IC50 = 2000 nM T64969 C4HNQ7 5328766 IC50 = 3100 nM T64969 CLQ73F 5328767 IC50 = 19054.61 nM T64969 C3F7YW 5328770 IC50 = 700 nM T64969 C67KXB 5328771 IC50 = 700 nM T64969 CJ6U2C 5328773 IC50 < 625 nM T64969 C7VW9X 5328774 IC50 = 2089.3 nM T64969 CSL05I 5328775 IC50 = 3000 nM T64969 C5ZV9K 5328776 IC50 = 1530 nM T64969 C3GRB0 5328777 IC50 = 1700 nM T64969 CI97TH 5328778 IC50 = 1700 nM T64969 CMX61C 5328780 IC50 = 4300 nM T64969 CED31Y 5328781 IC50 = 5100 nM T64969 CZ9Y4I 5328782 Ki = 240000 nM T64969 CBNU15 5328783 Ki = 150000 nM T64969 C2E4VB 5328784 Ki = 143000 nM T64969 CB2W9A 5328785 Ki = 49000 nM T64969 C75XMH 5328786 Ki = 24000 nM T64969 CH86SJ 5328787 Ki = 20000 nM T64969 CD8SN1 5328788 Ki = 10000 nM T64969 CJC2Z1 5328789 IC50 = 1300000 nM T64969 CF3MR6 5328790 IC50 = 264000 nM T64969 C94SUH 5328791 IC50 = 165000 nM T64969 C9PCS3 5328792 IC50 = 47000 nM T64969 C4N0CE 5328793 IC50 = 30000 nM T64969 CS98WX 5328794 IC50 > 1250000 nM T64969 CEA86M 5328795 Ki = 341000 nM T64969 CNB7Q3 5328796 IC50 = 800000 nM T64969 CGY6U3 5328797 Ki = 360000 nM T64969 CP50YI 5328798 IC50 = 500000 nM T64969 CD6JM3 5328799 IC50 = 450000 nM T64969 C5HQJ7 5328800 IC50 = 230000 nM T64969 CS09OR 5328801 Ki = 4500 nM T64969 CD6SC0 5328802 IC50 = 50000 nM T64969 C46UBD 5328805 IC50 = 60000 nM T64969 CR4K3Z 5328806 IC50 = 2500 nM T64969 CYO4C9 5328808 IC50 = 1000 nM T64969 CB8QZ6 5328809 IC50 = 500 nM T64969 C8M2UN 5328810 IC50 = 1360000 nM T64969 CLQA04 5328811 IC50 = 2400000 nM T64969 C5H3UK 5328812 Ki = 24000 nM T64969 CWJQ49 5328813 IC50 = 225000 nM T64969 C69RVL 5328814 IC50 = 350000 nM T64969 CU73YL 5328815 IC50 = 1400000 nM T64969 CEUV72 5328835 IC50 > 1000000 nM T64969 C2IN6M 5328838 IC50 = 416.87 nM T64969 CH6F9K 5328839 IC50 = 977.24 nM T64969 C7YRI8 5328840 IC50 = 90 nM T64969 CIQ54V 5328841 IC50 = 181.97 nM T64969 CCUR96 5328842 IC50 = 1445.44 nM T64969 CXH6C3 5328843 IC50 = 50118.72 nM T64969 CI9M3J 5328844 IC50 = 741.31 nM T64969 CB8RH3 5328845 IC50 = 14125.38 nM T64969 CJO6F4 5328846 IC50 = 47863.01 nM T64969 C2TQ4I 5328847 IC50 = 7413.1 nM T64969 C3QYM2 5328848 IC50 = 812.83 nM T64969 CU16VD 5328849 IC50 = 851.14 nM T64969 CX2CO0 5328850 IC50 = 870.96 nM T64969 CQK10C 5328851 IC50 = 5170 nM T64969 C0G6RT 5328852 IC50 = 13803.84 nM T64969 C9BYN7 5328853 IC50 = 6309.57 nM T64969 CZ3XY7 5328854 IC50 = 2754.23 nM T64969 C4K2ST 5328855 IC50 = 7762.47 nM T64969 CK6HN0 5328856 IC50 = 1778.28 nM T64969 CM60SD 5328857 IC50 = 9120.11 nM T64969 CL21YK 5328858 IC50 = 3162.28 nM T64969 CD1R8Q 5328859 IC50 = 16982.44 nM T64969 CY5MV7 5328860 IC50 = 758.58 nM T64969 C36EMZ 5328861 IC50 = 1479.11 nM T64969 CIXV80 5328863 IC50 = 229.09 nM T64969 CCE96Z 5328864 IC50 = 363.08 nM T64969 CMV0J2 5328865 IC50 = 61659.5 nM T64969 C47VGY 5328866 IC50 = 6606.93 nM T64969 CLOF23 5328867 IC50 = 4168.69 nM T64969 C3UBZ5 5328868 IC50 = 158.49 nM T64969 C5XM1A 5328869 IC50 = 831.76 nM T64969 C80RXA 5328870 IC50 = 616.6 nM T64969 C0KX1O 5328871 IC50 = 2187.76 nM T64969 CFIH48 5328872 IC50 = 69183.1 nM T64969 CBC41T 5328873 IC50 = 33113.11 nM T64969 CDG14R 5328874 IC50 = 21379.62 nM T64969 C5E0TK 5328877 IC50 = 3388.44 nM T64969 CC93DK 5328878 IC50 = 33884.42 nM T64969 C8F2JU 5328879 IC50 = 15135.61 nM T64969 C15RWZ 5328881 IC50 = 6760.83 nM T64969 CC3JI8 5328882 IC50 = 1096.48 nM T64969 CX18GK 5328883 IC50 = 6760.83 nM T64969 CYJ3W2 5328884 IC50 = 5128.61 nM T64969 CN5PO1 5328885 IC50 = 70794.58 nM T64969 C2PSJ1 5328886 IC50 = 89125.09 nM T64969 CT1QC6 5328954 IC50 = 6 nM T64969 C41BJK 5328955 IC50 = 12 nM T64969 CUW4V3 5328956 IC50 = 62 nM T64969 CI3Q6X 5328957 IC50 = 85 nM T64969 C0AF9T 5328958 IC50 = 97 nM T64969 C8A4XJ 5328959 IC50 = 71 nM T64969 CTN9X5 5328960 IC50 = 57 nM T64969 CP6G8R 5328961 IC50 = 20 nM T64969 CAQM41 5328962 IC50 = 95 nM T64969 CDJ8B5 5328964 IC50 = 65 nM T64969 C94KSU 5328965 IC50 = 9 nM T64969 C1W0DS 5328966 IC50 = 65 nM T64969 CX5S2M 5328967 IC50 = 59 nM T64969 CHL05B 5328968 IC50 = 2 nM T64969 CXN2Y0 5328969 IC50 = 0.22 nM T64969 C6BM9P 5328970 IC50 = 73 nM T64969 CR3GV8 5328971 IC50 = 90 nM T64969 CJU57A 5328972 IC50 = 106 nM T64969 CJ42FQ 5328973 IC50 = 74 nM T64969 CKA09Y 5328974 IC50 = 203 nM T64969 C92KTO 5328975 IC50 = 131 nM T64969 C4KI5U 5328976 IC50 = 85 nM T64969 CI36GZ 5328977 IC50 = 62 nM T64969 CU4W7S 5328978 IC50 = 14 nM T64969 C39VSH 5328979 IC50 = 68 nM T64969 C9U5YF 5328980 IC50 = 1124 nM T64969 CY4B5J 5328981 IC50 = 16 nM T64969 C03WIS 5328982 IC50 = 0.55 nM T64969 CG3KL4 5328983 IC50 = 1132 nM T64969 CV5KY4 5328984 IC50 = 115 nM T64969 CUJ6G5 5328985 IC50 = 107 nM T64969 CLP07T 5328986 IC50 = 250 nM T64969 CD60RC 5328987 IC50 = 215 nM T64969 CK15AU 5328988 IC50 = 269 nM T64969 C7R2EK 5328989 IC50 = 194 nM T64969 CFW19M 5329009 IC50 = 1 nM T64969 CZU0K3 5329011 IC50 = 100 nM T64969 C1XJL0 5329019 IC50 = 300 nM T64969 C9SZ4Q 5329020 IC50 = 100 nM T64969 C3VHF6 5329026 IC50 = 300 nM T64969 C9VX8C 5329040 IC50 = 1400 nM T64969 CK6T4U 5329042 IC50 = 400 nM T64969 CA81XO 5329045 IC50 = 450 nM T64969 C4T3MO 5329046 IC50 = 300 nM T64969 CQ15KR 5329049 IC50 = 450 nM T64969 C49KNS 5329050 IC50 = 500 nM T64969 C3C1EZ 5329051 IC50 = 400 nM T64969 C0H5XL 5329052 IC50 = 300 nM T64969 CW0KA8 5329053 IC50 = 200 nM T64969 COEN93 5329054 IC50 = 80 nM T64969 CATX52 5329055 IC50 = 100 nM T64969 CEQP41 5329056 IC50 = 150 nM T64969 CDV4C9 5329057 IC50 = 100 nM T64969 CH26SN 5329069 IC50 = 0.91 nM T64969 C7RF9L 5329070 IC50 = 0.17 nM T64969 CGTA78 5329071 IC50 = 1.6 nM T64969 CBV46K 5329072 IC50 = 0.5 nM T64969 CXG29Q 5329074 IC50 = 1.75 nM T64969 C6MX8O 5329075 IC50 = 27 nM T64969 CN02JA 5329077 IC50 = 9.1 nM T64969 CF0U7Z 5329078 IC50 = 1039 nM T64969 CE0UT9 5329079 IC50 = 0.37 nM T64969 CJFE40 5329080 IC50 = 2.7 nM T64969 CS84JW 5329081 IC50 = 1.5 nM T64969 C71GUX 5329082 IC50 = 4.2 nM T64969 C07AVK 5329083 IC50 = 2.7 nM T64969 CHS1I6 5329084 IC50 = 3.3 nM T64969 C5JL2Y 5329085 IC50 = 2.4 nM T64969 CT4U5F 5329086 IC50 = 0.44 nM T64969 CBY4R5 5329087 IC50 = 1.1 nM T64969 C53HOJ 5329088 IC50 = 0.73 nM T64969 C2P3EO 5329089 IC50 = 0.81 nM T64969 C61NGH 5329090 IC50 = 14 nM T64969 CUZ82W 5329091 IC50 = 1.45 nM T64969 CAV71E 5329092 IC50 = 0.6026 nM T64969 C0OD8J 5329093 IC50 = 0.76 nM T64969 C0A8HY 5329094 IC50 = 2.7 nM T64969 CPH8Q3 5329095 IC50 = 93.5 nM T64969 CG2QX5 5329096 IC50 = 0.4266 nM T64969 CE48UM 5329097 IC50 = 340 nM T64969 C9I7WT 5329100 IC50 > 20000 nM T64969 CMWB28 5329101 IC50 > 20000 nM T64969 CGX50J 5329104 IC50 = 10000 nM T64969 C2VX0H 5329105 IC50 > 20000 nM T64969 CK71MQ 5329106 IC50 > 20000 nM T64969 C6YRH8 5329108 IC50 > 20000 nM T64969 CFP59Y 5329109 IC50 > 20000 nM T64969 CSY10K 5329111 IC50 = 5530 nM T64969 C0JW3Y 5329134 IC50 = 28800 nM T64969 CO7J2A 5329135 IC50 > 50000 nM T64969 CQ4TP5 5329136 IC50 = 49200 nM T64969 CXQC42 5329137 IC50 > 50000 nM T64969 CT94JS 5329138 IC50 > 50000 nM T64969 CNH06M 5329139 IC50 > 100000 nM T64969 CRY4Z2 5329140 IC50 > 50000 nM T64969 CAPE50 5329141 IC50 > 50000 nM T64969 CFU58A 5329142 IC50 = 21800 nM T64969 C5Q8XK 5329143 IC50 = 30500 nM T64969 C8PX4D 5329144 IC50 = 19200 nM T64969 C6USQ5 5329145 IC50 = 22800 nM T64969 C56LWT 5329146 IC50 > 100000 nM T64969 CZ16MN 5329147 IC50 > 50000 nM T64969 CAN16I 5329148 IC50 > 50000 nM T64969 CG4NC2 5329149 IC50 > 100000 nM T64969 CIW70H 5329150 IC50 = 21900 nM T64969 C5FT6A 5329151 IC50 = 24100 nM T64969 CB0N4L 5329152 IC50 = 31300 nM T64969 COFP24 5329153 IC50 > 50000 nM T64969 CGWD98 5329154 IC50 > 100000 nM T64969 C4PD0K 5329156 IC50 > 100000 nM T64969 C0RWT8 5329157 IC50 > 100000 nM T64969 C3MU5S 5329158 IC50 > 100000 nM T64969 CN6O4R 5329159 IC50 > 100000 nM T64969 CG68DI 5329160 IC50 > 100000 nM T64969 CYR7V0 5329161 IC50 > 100000 nM T64969 C9BXE2 5329162 IC50 > 100000 nM T64969 CY4V5Z 5329163 IC50 > 100000 nM T64969 CI64YA 5329164 IC50 > 100000 nM T64969 C2ZV0O 5329165 IC50 = 29100 nM T64969 CAB53L 5329166 IC50 = 56500 nM T64969 CTW9R8 5329167 IC50 > 100000 nM T64969 C8A3TJ 5329168 IC50 > 100000 nM T64969 CVTD82 5329169 IC50 = 8880 nM T64969 CQ5WK1 5329170 IC50 > 100000 nM T64969 CNC9T7 5329171 IC50 > 100000 nM T64969 C6L0UW 5329229 IC50 > 20000 nM T64969 C1DBV6 5329230 IC50 = 180 nM T64969 CLKM80 5329231 IC50 = 200 nM T64969 CTQ18A 5329232 IC50 = 7820 nM T64969 CM5KG6 5329233 IC50 = 4.7 nM T64969 CQG6R2 5329234 IC50 = 29 nM T64969 CJ3A9I 5329235 IC50 = 22 nM T64969 CPS7X1 5329236 IC50 = 6.5 nM T64969 CAN60T 5329237 IC50 > 20000 nM T64969 CY15JP 5329238 IC50 = 5310 nM T64969 C41UBI 5329239 IC50 = 40 nM T64969 C6VQ9F 5329240 IC50 = 2.8 nM T64969 C8WS5K 5329241 IC50 = 210 nM T64969 CI26UN 5329242 IC50 = 410 nM T64969 C6PJ2R 5329243 IC50 = 13 nM T64969 C0OKB7 5329244 IC50 = 200 nM T64969 C78ZNL 5329245 IC50 = 5.9 nM T64969 CWL5S4 5329246 IC50 = 0.45 nM T64969 C4X3OE 5329248 IC50 = 450 nM T64969 CK8FH6 5329249 IC50 = 1410 nM T64969 CN5B6C 5329250 IC50 = 100 nM T64969 CQ0B6E 5329251 IC50 = 100 nM T64969 C4KO3N 5329252 IC50 = 200 nM T64969 C6MZF8 5329253 IC50 > 20000 nM T64969 CO1U8I 5329254 IC50 = 340 nM T64969 C54NXZ 5329255 IC50 = 400 nM T64969 CN4MD2 5329256 IC50 = 10000 nM T64969 CJ9O8L 5329257 IC50 = 4300 nM T64969 C0WJ6Y 5329258 IC50 = 5000 nM T64969 CA6H2Y 5329259 IC50 = 700 nM T64969 CFP2O6 5329260 IC50 = 700 nM T64969 CV6KI2 5329261 IC50 = 1300 nM T64969 CLK4V3 5329262 IC50 = 6000 nM T64969 CXUV69 5329263 IC50 = 12500 nM T64969 CSV71T 5329264 IC50 = 19000 nM T64969 C9S6OV 5329266 IC50 = 2200 nM T64969 CIV10W 5329267 IC50 = 2200 nM T64969 C96PSZ 5329268 IC50 = 4000 nM T64969 CJR4T0 5329269 IC50 > 100000 nM T64969 CP20TG 5329270 IC50 = 2000 nM T64969 C8R2YT 5329271 IC50 = 1400 nM T64969 C2AR4T 5329272 IC50 = 940 nM T64969 CD6NV0 5329475 IC50 = 34.67 nM T64969 CA78HB 5329476 IC50 = 81.28 nM T64969 C0OAR2 5329477 IC50 = 70.79 nM T64969 C8A3GZ 5329478 IC50 = 537.03 nM T64969 C78XVZ 5329479 IC50 = 7.943 nM T64969 CQ39FM 5329480 IC50 = 10 nM T64969 CVS3Z1 5329481 IC50 = 97.72 nM T64969 CW2UJ7 5329482 IC50 = 263 nM T64969 CY14AK 5329483 IC50 = 74 nM T64969 CIT24W 5329484 IC50 = 68 nM T64969 CDZ6R5 5329485 IC50 = 79 nM T64969 C3LSH8 5329486 IC50 = 104 nM T64969 CGZA12 5329487 IC50 = 830 nM T64969 CV9L1J 5329488 IC50 = 74.13 nM T64969 CJD92I 5329489 IC50 = 11 nM T64969 CS1HF6 5329490 IC50 = 19.95 nM T64969 CX4L0Q 5329491 IC50 = 93 nM T64969 C9C3SD 5329492 IC50 = 27 nM T64969 CDRM58 5329493 IC50 = 24 nM T64969 CS2HM9 5329714 IC50 > 50000 nM T64969 CM9V8E 5329715 IC50 > 50000 nM T64969 CB0QZ2 5330117 IC50 > 1000 nM T64969 C7QZL3 5330118 IC50 > 1000 nM T64969 CNR9B8 5330119 IC50 > 1000 nM T64969 CXY2I9 5330120 IC50 > 1000 nM T64969 CDF96J 5330121 IC50 > 1000 nM T64969 C7BPR2 5330122 IC50 > 1000 nM T64969 CC4ZJ3 5330123 IC50 > 1000 nM T64969 CLV0T6 5330124 IC50 > 1000 nM T64969 CZ3LK2 5330387 IC50 = 1360 nM T64969 CRU94N 5330388 IC50 = 7400 nM T64969 CDB68F 5330389 IC50 > 10000 nM T64969 C7CX0H 5330390 IC50 > 10000 nM T64969 C5SY4O 5330420 IC50 = 2000 nM T64969 CUEZ35 5330437 IC50 = 2700 nM T64969 C94GRU 5330453 IC50 = 3000 nM T64969 CC2E4Q 5330468 IC50 = 7100 nM T64969 C1YWE0 5330475 IC50 = 27000 nM T64969 C9NBG7 5330546 IC50 > 10000 nM T64969 CF01JS 5330804 IC50 = 8400 nM T64969 C3U0TG 5330830 IC50 > 100000 nM T64969 CL1FH5 5330832 IC50 > 100000 nM T64969 C1P2ZA 5330847 IC50 > 100000 nM T64969 CM47KI 5351344 IC50 > 10000 nM T64969 CYXI29 5353388 IC50 = 400 nM T64969 CJ5A1W 5353391 IC50 = 100 nM T64969 CHD1L6 5353609 IC50 = 20 ug.mL-1 T64969 CQ12UT 5353911 IC50 = 0.1 ug.mL-1 T64969 CDQ3M7 5359485 IC50 = 5.5 ug.mL-1 T64969 C54BYP 5360741 IC50 = 1.7 ug.mL-1 T64969 C6REP3 5371842 IC50 = 38460 nM T64969 CB8DX4 5371857 IC50 = 29850 nM T64969 C23XEH 5386499 IC50 > 100 ug.mL-1 T64969 CL5W9P 5386517 IC50 > 10 ug.mL-1 T64969 C63YGX 5386800 IC50 = 0.3 ug.mL-1 T64969 C0SO6F 5388678 IC50 = 10000 nM T64969 C6RAT9 5388682 IC50 = 7000 nM T64969 C2O9ZG 5391486 IC50 = 31800 nM T64969 CD65JT 5427216 IC50 > 100000 nM T64969 CPB95V 5427224 IC50 > 100000 nM T64969 CL27VO 5467485 IC50 = 20300 nM T64969 CRKI23 5468831 IC50 = 5800 nM T64969 CZ0NU2 5481591 IC50 > 1000 nM T64969 CCT39K 5703472 IC50 = 10100 nM T64969 CA6L5V 5707304 IC50 > 100000 nM T64969 C43YGE 5713379 IC50 > 100000 nM T64969 CS24NJ 5775636 IC50 = 9000 nM T64969 CT8U7I 5874584 IC50 > 100000 nM T64969 CO6KI2 5930298 IC50 > 10000 nM T64969 CRW23P 5941457 IC50 = 400 nM T64969 CM8LW9 6036100 IC50 > 100000 nM T64969 CPU89Q 6082393 IC50 = 35000 nM T64969 C7MD9J 6091659 IC50 = 18600 nM T64969 C3R9VW 6105823 IC50 = 3 ug.mL-1 T64969 C9XV5P 6398579 IC50 = 1300000 nM T64969 C0IYS8 6408948 IC50 = 76 nM T64969 C18VEH 6415635 IC50 = 65 nM T64969 C0ITJ4 6419347 IC50 = 4.1 nM T64969 C61JMS 6419746 IC50 = 440000 nM T64969 CZF6Y9 6439072 IC50 = 1000 nM T64969 CO5SZ1 6440837 IC50 > 200 ug.mL-1 T64969 C4KVL5 6441269 IC50 = 19000000 nM T64969 C83XSI 6442618 IC50 = 8 ug.mL-1 T64969 C9YRT1 6447922 IC50 = 4000 nM T64969 CXO27Z 6447923 IC50 = 20000 nM T64969 CTB7N5 6447926 IC50 = 398.11 nM T64969 C49YOE 6447934 IC50 = 3000 nM T64969 CQ3S8L 6450842 IC50 > 100000 nM T64969 C2N0IR 6477203 IC50 > 50000 nM T64969 CL8MC2 6505651 IC50 > 10 ug.mL-1 T64969 CW5YJ2 6536705 IC50 > 100000 nM T64969 C0O8DH 6538899 IC50 = 1680 nM T64969 CUPQ08 6539985 IC50 > 50000 nM T64969 CMEZ23 6540005 IC50 > 50000 nM T64969 CP0XI6 6603792 IC50 = 177 nM T64969 CUJ97R 7023155 IC50 = 6800 nM T64969 C0MGV7 7048595 IC50 = 2800 nM T64969 C14UAT 7574840 IC50 > 10000 nM T64969 CV7L5M 8895911 IC50 > 10000 nM T64969 CY01OB 9209612 IC50 = 57000 nM T64969 CH46ZU 9583801 IC50 > 100000 nM T64969 C4A8RX 9794758 IC50 = 510 nM T64969 C2OL7K 9796455 IC50 = 3700 nM T64969 CZR3M4 9799152 IC50 > 100000 nM T64969 C2B4ZE 9803006 IC50 = 910 nM T64969 CF47BP 9806229 IC50 = 0.79 nM T64969 C72WMK 9808725 IC50 = 91 nM T64969 CZ2MH9 9809611 IC50 = 19 nM T64969 CI3O6X 9814609 IC50 > 100000 nM T64969 CUNV09 9816954 IC50 = 27000 nM T64969 CK2DM9 9818251 IC50 = 100 nM T64969 C4Z2GW 9819930 IC50 = 797 nM T64969 CZ5VX6 9820644 IC50 = 0.2512 nM T64969 CKR04B 9821918 IC50 = 700 nM T64969 CX9DG5 9822042 IC50 > 100000 nM T64969 CRKD07 9825976 IC50 = 33 nM T64969 C1E2DV 9826083 IC50 = 8700 nM T64969 C9TAL6 9826308 IC50 > 48000 nM T64969 C4XU5Z 9828336 IC50 = 27 nM T64969 C5S8FR 9829680 IC50 = 28 nM T64969 CYWI50 9830092 IC50 = 160 nM T64969 CBGE59 9833337 IC50 = 2000 nM T64969 CFPI31 9844683 IC50 = 3200 nM T64969 CSH0A9 9847014 IC50 = 530 nM T64969 CGKC15 9851149 IC50 = 100 nM T64969 C41QWA 9857146 IC50 = 6300 nM T64969 C43FVO 9859850 IC50 = 340 nM T64969 C3UQL7 9860872 IC50 = 100000 nM T64969 C16VXB 9863538 IC50 > 10000 nM T64969 CW8V0K 9864418 IC50 > 25000 nM T64969 CGC0F7 9864462 IC50 = 2.5 nM T64969 CTN7L4 9869773 IC50 = 200 nM T64969 CM5Z8X 9869943 IC50 > 10000 nM T64969 C12PKF 9871380 IC50 = 40 nM T64969 C2FW1X 9872621 IC50 = 18 nM T64969 CS51KJ 9873631 IC50 = 43 nM T64969 CU2N8D 9873657 IC50 = 18 nM T64969 C5NK9U 9873849 IC50 = 27 nM T64969 C5CLD8 9874613 IC50 = 90 nM T64969 CM2QX5 9879615 IC50 = 4100 nM T64969 CSB5D8 9882519 IC50 = 200 nM T64969 CY70OD 9882602 IC50 = 6 nM T64969 CPJ7W2 9882655 IC50 > 20000 nM T64969 CV1A2S 9883384 IC50 = 170 nM T64969 CE47IF 9884465 IC50 = 3 nM T64969 C4R8YV 9884654 IC50 = 1 nM T64969 CUZ07T 9884745 IC50 = 7900 nM T64969 CL5BD2 9885081 IC50 = 39 nM T64969 C2JR8Q 9887521 IC50 = 933.25 nM T64969 CR2B8U 9888491 IC50 = 1704 nM T64969 CXL31W 9890154 IC50 = 2320 nM T64969 CHF7G5 9890746 IC50 > 100000 nM T64969 CIN0E2 9891993 IC50 = 13489.63 nM T64969 CXA5C8 9893493 IC50 = 4200 nM T64969 CE87TX 9893671 IC50 = 24 nM T64969 CEJ05V 9894581 IC50 = 26 nM T64969 C4WQK8 9897300 IC50 = 3.6 nM T64969 CB4DT1 9899125 IC50 = 5600 nM T64969 CP04SA 9906350 IC50 = 10000 nM T64969 C01WSX 9907221 IC50 = 1.6 nM T64969 CO7RU2 9908666 IC50 = 0.4 nM T64969 C2TC1L 9910609 IC50 = 239 nM T64969 C3EUB4 9911005 IC50 > 100000 nM T64969 C9SQU4 9913648 IC50 = 1600 nM T64969 C5GE7T 9917045 IC50 = 5400 nM T64969 CF3KI0 9917474 IC50 = 25 nM T64969 C2DL8U 9927208 IC50 = 4 nM T64969 CYW49X 9927718 IC50 = 10000 nM T64969 CG6A1H 9927800 IC50 > 10000 nM T64969 CWT56C 9930439 IC50 = 86.9 nM T64969 CP2J4W 9930632 IC50 = 3.6 nM T64969 CPYB98 9934935 IC50 = 1910293.07 nM T64969 CU56DE 9937225 IC50 = 23 nM T64969 CLT0U5 9937660 IC50 = 12 nM T64969 CXJR73 9938805 IC50 = 89 nM T64969 CUKH27 9943194 IC50 = 50000 nM T64969 CU78NO 9947433 IC50 > 100000 nM T64969 CYI65J 9948215 IC50 = 29 nM T64969 C6HP3L 9948410 IC50 > 100000 nM T64969 C0U6EJ 9949448 IC50 > 100000 nM T64969 C06JHE 9952784 IC50 = 0.07 nM T64969 CYT7R9 9953676 IC50 > 100000 nM T64969 CI51BV 9954075 IC50 = 645.65 nM T64969 CBE9O6 9954156 IC50 = 36 nM T64969 CJM8R9 9956715 IC50 = 1000 nM T64969 C0ZO2V 9960493 IC50 = 21 nM T64969 CSU19Y 9960734 IC50 = 85 nM T64969 CJ40GO 9965429 IC50 > 100000 nM T64969 CIKN68 9965616 IC50 = 2 ug.mL-1 T64969 CAH50Y 9970231 IC50 = 14100 nM T64969 CM8NB2 9972089 IC50 > 20000 nM T64969 C24MZU 9974694 IC50 = 3.1 nM T64969 CZN09Q 9977010 IC50 > 1000 nM T64969 CCV62S 9978638 IC50 = 1500 nM T64969 CROV41 9979362 IC50 = 850 nM T64969 C6BXQ9 9979953 IC50 = 5000 nM T64969 CA6Z4L 9980337 IC50 = 5000 nM T64969 CFVI29 9981239 IC50 = 8.6 nM T64969 CB2KF5 9981727 IC50 = 35 nM T64969 C37GXK 9983303 IC50 > 25000 nM T64969 CH03DY 9984664 IC50 = 10320 nM T64969 C29SOH 9985870 IC50 > 100000 nM T64969 CQZF34 9994794 IC50 > 100000 nM T64969 CO4N3Q 9995374 IC50 > 100000 nM T64969 CFG0E8 9996177 IC50 = 20000 nM T64969 CF0SE3 9998325 IC50 = 900 nM T64969 CMYI47 10002824 IC50 = 2 nM T64969 CNY2F1 10005402 IC50 = 2 nM T64969 C26QHZ 10005638 IC50 > 10000 nM T64969 CQX39R 10006530 IC50 = 80 nM T64969 C0EWK9 10007087 IC50 = 10000 nM T64969 CH7DN2 10009462 IC50 = 16900 nM T64969 CF2V4B 10016116 IC50 > 10000 nM T64969 C7WJ5H 10016952 IC50 = 66100 nM T64969 CWH02V 10018196 IC50 > 20000 nM T64969 CA5E4R 10019589 IC50 = 1000 nM T64969 C86HYI 10020830 IC50 = 70 nM T64969 C53UTR 10022185 IC50 = 8800 nM T64969 C1Y0PX 10023383 IC50 < 5 nM T64969 CO2PA9 10029703 IC50 = 5390 nM T64969 C19XDW 10032479 IC50 > 100000 nM T64969 C0IA4P 10037831 IC50 = 8700 nM T64969 CXL0R8 10038606 IC50 > 100000 nM T64969 CD4Z1B 10040645 IC50 = 9500 nM T64969 C8TY1B 10040646 IC50 = 3000 nM T64969 C2M8VJ 10040715 IC50 > 20000 nM T64969 C8VNJ1 10041429 IC50 = 37500 nM T64969 C0XAV7 10041970 IC50 = 3000 nM T64969 CE98SN 10041980 IC50 > 20000 nM T64969 C1YV0B 10043236 IC50 = 100 nM T64969 C8IS1F 10043899 IC50 = 400 nM T64969 C25JLD 10043994 IC50 = 2000 nM T64969 CF03ZB 10044469 IC50 = 90 nM T64969 CAZ71W 10045755 IC50 ~ 4000 nM T64969 CJ6L3T 10046873 IC50 > 50000 nM T64969 CG57EC 10047098 IC50 = 300 nM T64969 C7YD1X 10048045 IC50 > 25000 nM T64969 C54AEL 10048519 IC50 = 2100 nM T64969 C9VQZ3 10053637 IC50 = 47000 nM T64969 CFS2H4 10053638 IC50 > 100000 nM T64969 C32WOU 10058766 IC50 > 20000 nM T64969 C6K0XB 10064040 IC50 = 670 nM T64969 CR7TY8 10064290 IC50 > 20000 nM T64969 C5UPR6 10065338 IC50 = 6.4 nM T64969 CBF54I 10066030 IC50 = 8700 nM T64969 C82XJV 10067396 IC50 = 80 nM T64969 CH2WO5 10067548 IC50 = 490 nM T64969 C2L3JB 10068026 IC50 = 6900 nM T64969 C0DR5I 10068517 IC50 = 0.6761 nM T64969 C7DNB8 10070557 IC50 = 21 nM T64969 CCK25W 10070969 IC50 = 45800 nM T64969 CK8RL4 10071409 IC50 = 125 ug.mL-1 T64969 C7J8YN 10073101 IC50 = 8800 nM T64969 C1JUF8 10073832 IC50 > 10000 nM T64969 CF1D6Y 10075240 IC50 > 10000 nM T64969 CC0J9E 10075664 IC50 = 25 nM T64969 CD5B6O 10076837 IC50 > 100000 nM T64969 CMK64J 10084671 IC50 = 21000 nM T64969 C8A1TH 10085171 IC50 > 100000 nM T64969 CM96YH 10085557 IC50 = 600 nM T64969 C2C1BP 10089048 IC50 > 25000 nM T64969 C8HEJ2 10092460 IC50 = 800 nM T64969 COW60X 10092803 IC50 = 400 nM T64969 CX6N2G 10092804 IC50 = 360 nM T64969 CH62FG 10093300 IC50 = 7000 nM T64969 CF09NK 10098235 IC50 = 3830 nM T64969 CK50LJ 10100761 IC50 = 47000 nM T64969 C10SZX 10106602 IC50 > 20000 nM T64969 CZ9Y1G 10106867 IC50 = 11 nM T64969 C3P8WK 10110378 IC50 > 100000 nM T64969 C63CFD 10111108 IC50 > 100000 nM T64969 C7TA9J 10113568 IC50 = 10000 nM T64969 C5SV9C 10114464 IC50 = 64 nM T64969 C80ZDK 10115240 IC50 = 90 nM T64969 C7C1IG 10116123 IC50 = 110 nM T64969 CMK79O 10117051 IC50 = 200 nM T64969 CYV4I1 10127271 IC50 = 9300 nM T64969 CA31MX 10131256 IC50 = 650 nM T64969 CV4QA0 10136035 IC50 = 4800 nM T64969 C53JSE 10136105 IC50 = 680 nM T64969 CL42XS 10136330 IC50 > 100000 nM T64969 CREM37 10151881 IC50 = 35 nM T64969 CC4X6M 10152238 IC50 = 5 nM T64969 C5HB2P 10152514 IC50 = 48 nM T64969 C14ZEP 10156890 IC50 = 1061 nM T64969 CUW34X 10157645 IC50 = 100000 nM T64969 CUD7L1 10159833 IC50 = 45 nM T64969 CZE4S6 10159951 IC50 = 10 nM T64969 CA40TZ 10161969 IC50 = 790 nM T64969 CHU9C6 10162630 IC50 = 690 nM T64969 CK4OH0 10162954 IC50 = 698 nM T64969 CGW26V 10163178 IC50 = 0.5 nM T64969 C9LH1R 10172616 IC50 = 720 nM T64969 CZ4X7O 10172837 IC50 > 10000 nM T64969 CC56EH 10173248 IC50 = 10 nM T64969 CC78NE 10179293 IC50 = 853 nM T64969 C6H3FI 10180188 IC50 = 21 nM T64969 COC30E 10181160 IC50 > 100000 nM T64969 C3GFB0 10194325 IC50 = 55 nM T64969 CNYA34 10194617 IC50 = 9000 nM T64969 CQP8Y1 10194801 IC50 = 90 nM T64969 CI4Q0J 10195479 IC50 = 73 nM T64969 C1TX8D 10198953 IC50 = 29400 nM T64969 C2RLF5 10199254 IC50 = 200 nM T64969 C47FXG 10200918 IC50 = 1139 nM T64969 CGOT91 10207821 IC50 > 100000 nM T64969 C5YCN2 10215023 IC50 > 100000 nM T64969 CZ0XD7 10215809 IC50 = 390 nM T64969 CP81YE 10216042 IC50 = 2 nM T64969 CVQ53X 10216257 IC50 = 560 nM T64969 C36YTW 10216482 IC50 = 45 nM T64969 CZ2A0F 10216910 IC50 = 5 nM T64969 CNTU23 10217083 IC50 = 60 nM T64969 CSGL59 10217304 IC50 = 170 nM T64969 CEW30I 10217590 IC50 = 61 nM T64969 C74AGX 10222656 IC50 = 71 nM T64969 C67POS 10223065 IC50 = 1620 nM T64969 CCVU79 10226418 IC50 = 160 nM T64969 C2KSD3 10227095 IC50 = 350 nM T64969 C6QP4E 10227907 IC50 = 63 nM T64969 CD7J3O 10231458 IC50 > 30000 nM T64969 CPD6Z9 10236164 IC50 > 100000 nM T64969 CV7PU8 10237247 IC50 = 85 nM T64969 C0UN1C 10245626 IC50 > 20000 nM T64969 CQ3LT1 10245856 IC50 = 14 nM T64969 CSGD16 10246246 IC50 > 7000 nM T64969 CYMD04 10246609 IC50 > 20000 nM T64969 CLV83M 10246831 IC50 > 50000 nM T64969 CU53QW 10247949 IC50 = 5000 nM T64969 CGME21 10248155 IC50 > 100000 nM T64969 C97GRN 10248747 IC50 = 100000 nM T64969 CNH85V 10249869 IC50 = 1300 nM T64969 CC9E5Q 10249989 IC50 > 10000 nM T64969 C1WL8B 10251852 IC50 = 22800 nM T64969 CH30RC 10253133 IC50 > 10000 nM T64969 C1UB5A 10253204 IC50 = 309.03 nM T64969 C32KTH 10253992 IC50 = 21200 nM T64969 CG2TF7 10255849 IC50 = 7700 nM T64969 CBR9P3 10257058 IC50 = 17500 nM T64969 C6G8NR 10264200 IC50 > 100000 nM T64969 C3HF6S 10264201 IC50 > 100000 nM T64969 CBI47E 10264222 IC50 > 100000 nM T64969 CF81EM 10265006 IC50 > 100000 nM T64969 CHFZ23 10266516 IC50 = 180 nM T64969 CWY4U3 10267270 IC50 = 460 nM T64969 CJGH26 10275985 IC50 = 2290 nM T64969 C6PL7V 10276061 IC50 = 64 nM T64969 CY67TW 10287149 IC50 = 11 nM T64969 C4W6JL 10287402 IC50 = 18 nM T64969 CT3W9O 10287552 IC50 = 2 nM T64969 CE7Q8U 10288283 IC50 = 8 nM T64969 C9K0SA 10288761 IC50 = 140 nM T64969 CJ4D9B 10288917 IC50 = 240 nM T64969 CNU74Z 10288918 IC50 = 780 nM T64969 CCE64Z 10288920 IC50 = 35 nM T64969 CN51JQ 10292737 IC50 > 100000 nM T64969 C3FL9K 10295633 IC50 = 4400 nM T64969 C8NMA6 10295839 IC50 = 810 nM T64969 C7SFI1 10296883 IC50 > 10000 nM T64969 CVO54Z 10300451 IC50 = 40 nM T64969 C8RD3V 10301884 IC50 = 900 nM T64969 C1AKH9 10303277 IC50 > 1000 nM T64969 CY0A3T 10309300 IC50 = 3 nM T64969 C8DQ9O 10309491 IC50 = 1100 nM T64969 C3MJB0 10309561 IC50 = 11 nM T64969 CGF21D 10310843 IC50 = 68 nM T64969 C0SY1J 10314618 IC50 > 20000 nM T64969 CD34UM 10317124 IC50 = 2500 nM T64969 CW85MK 10317696 IC50 = 4000 nM T64969 CM1X0V 10318022 IC50 = 174 nM T64969 C39YNC 10318148 IC50 > 100000 nM T64969 C1KFM8 10318154 IC50 = 230 nM T64969 CK83IU 10318851 IC50 = 110 nM T64969 C27CDR 10319118 IC50 = 7300 nM T64969 CUC58I 10320940 IC50 = 0.12 nM T64969 CEN48D 10322889 IC50 = 790 nM T64969 CN23SU 10324074 IC50 > 1000 nM T64969 C6WJB8 10325906 IC50 > 50000 nM T64969 CCK42E 10327195 IC50 = 5300 nM T64969 CX7NM0 10327196 IC50 > 100000 nM T64969 CQ03XB 10327197 IC50 > 100000 nM T64969 COB74A 10330538 IC50 > 20000 nM T64969 CG1AS6 10333483 IC50 = 20000 nM T64969 COC7P1 10333957 IC50 > 100000 nM T64969 CQ80HY 10337047 IC50 = 1100 nM T64969 CET21U 10337153 IC50 = 1100 nM T64969 C9GK3M 10342546 IC50 = 1000 nM T64969 CU8LT7 10345125 IC50 > 50000 nM T64969 CD2H0G 10347728 IC50 = 43000 nM T64969 CNJ97S 10348925 IC50 = 5500 nM T64969 CZ0UL8 10349829 IC50 = 13000 nM T64969 CYCM39 10355659 IC50 > 100000 nM T64969 C37AMD 10356450 IC50 > 100000 nM T64969 C4DOQ9 10356451 IC50 = 7800 nM T64969 CE08LX 10356808 IC50 = 6000 nM T64969 CYI4N2 10357604 IC50 = 400 nM T64969 CT19AL 10359253 IC50 = 27500 nM T64969 C19VUI 10360971 IC50 > 50000 nM T64969 C3L5UZ 10361853 IC50 > 50000 nM T64969 C8RW0D 10362209 IC50 = 20 nM T64969 CD1R3L 10362325 IC50 = 200 nM T64969 C8H1OJ 10371203 IC50 = 1700 nM T64969 C7ACN5 10383837 IC50 = 700 nM T64969 CVP85S 10385997 IC50 = 10000 nM T64969 C6ZF0X 10386217 IC50 > 100000 nM T64969 C36GIL 10386874 IC50 = 4700 nM T64969 CQB9H7 10389422 IC50 = 4800 nM T64969 CA8B5T 10390073 IC50 = 1100 nM T64969 CQIK61 10406106 IC50 = 900 nM T64969 CF74ID 10406267 IC50 = 2500 nM T64969 CBMW34 10406907 IC50 > 20000 nM T64969 C34JQT 10407176 IC50 > 100000 nM T64969 C4SGL2 10407341 IC50 > 100000 nM T64969 CC13FP 10408738 IC50 = 90 nM T64969 C9RCU7 10408993 IC50 = 470 nM T64969 C4PV3R 10409198 IC50 = 5600 nM T64969 C32REN 10411907 IC50 = 4 nM T64969 CFJ2S1 10413621 IC50 >> 5000 nM T64969 CHPR58 10416818 IC50 = 12000 nM T64969 CVK10W 10421743 IC50 > 20000 nM T64969 CP6N2J 10423146 IC50 > 100000 nM T64969 C4T5WG 10424297 IC50 = 400 nM T64969 CHID58 10425395 IC50 > 20000 nM T64969 CQ43JU 10426229 IC50 = 400 nM T64969 CQR85O 10427421 IC50 > 20000 nM T64969 C7HBP6 10429593 IC50 > 10000 nM T64969 CE6P0T 10429844 IC50 = 50 nM T64969 C2SXE3 10430383 IC50 = 1000 nM T64969 CP14EC 10430484 IC50 = 3400 nM T64969 C3MI7D 10430804 IC50 = 300 nM T64969 CFLH53 10432113 IC50 = 800 nM T64969 C56SVY 10434122 IC50 = 1250 nM T64969 CN5BF4 10434923 IC50 = 50000 nM T64969 C7QU9X 10437879 IC50 > 100000 nM T64969 CXA85V 10439212 IC50 = 6100 nM T64969 CQHS12 10445612 IC50 > 25000 nM T64969 CEU25H 10445729 IC50 > 100000 nM T64969 C9XLN7 10446123 IC50 = 5400 nM T64969 C3LY4K 10447743 IC50 = 300 nM T64969 CUX75O 10450005 IC50 > 50000 nM T64969 CT42KE 10450849 IC50 > 100000 nM T64969 CL7PF2 10451087 IC50 = 3400 nM T64969 C9GJZ5 10453233 IC50 = 1000 nM T64969 CZ09AI 10454066 IC50 = 2700 nM T64969 CSZ40F 10455755 IC50 = 1250 nM T64969 C95LYF 10457505 IC50 > 100000 nM T64969 CYF3P4 10468511 IC50 = 9000 nM T64969 CW23SQ 10468973 IC50 > 100000 nM T64969 C2CVB8 10470221 IC50 > 100000 nM T64969 C4DTZ5 10470384 IC50 > 20000 nM T64969 CH4CY9 10471016 IC50 = 700 nM T64969 CI7BO0 10471069 IC50 = 7000 nM T64969 C3JIZ2 10473386 IC50 > 20000 nM T64969 CC5OM4 10473589 IC50 > 200 ug.mL-1 T64969 C5PAU6 10475547 IC50 = 100000 nM T64969 CC98AG 10475666 IC50 = 3000 nM T64969 C1GKT0 10476486 IC50 = 1000 nM T64969 CZ45NX 10476762 IC50 > 100000 nM T64969 CR07PO 10477008 IC50 = 700 nM T64969 CM9F3D 10477397 IC50 > 1000 nM T64969 C7PLI5 10478569 IC50 > 10000 nM T64969 CRX6F0 10479082 IC50 > 25000 nM T64969 COW2Q5 10483554 IC50 > 100000 nM T64969 CD7XE3 10484487 IC50 > 100000 nM T64969 CJWH60 10489322 IC50 > 100000 nM T64969 C0EV8B 10494548 IC50 = 6000 nM T64969 C05ANY 10494804 IC50 = 538 nM T64969 CZ06SL 10495153 IC50 > 100000 nM T64969 C8DH5W 10499619 IC50 = 12500 nM T64969 C78FPR 10501266 IC50 = 1800 nM T64969 C1O6YQ 10502559 IC50 > 50000 nM T64969 CB76HG 10504176 IC50 = 2 nM T64969 C3DK8I 10520057 IC50 = 0.25 nM T64969 CB3MW7 10522352 IC50 = 0.91 nM T64969 C7RFN2 10523147 IC50 = 1.1 nM T64969 CLH12I 10523411 IC50 = 291 nM T64969 C0GP2I 10523766 IC50 > 5000 nM T64969 C38RSF 10528818 IC50 = 0.16 nM T64969 CBC2E1 10530118 IC50 = 3 nM T64969 C5SVT4 10537949 IC50 > 100000 nM T64969 CU0E9F 10538285 IC50 = 6920 nM T64969 C3VPC7 10538965 IC50 > 100000 nM T64969 CG63KU 10539833 IC50 = 1200 nM T64969 CXT20A 10541248 IC50 = 500 nM T64969 C8VJX1 10542530 IC50 > 5000 nM T64969 C7JX3G 10547930 IC50 = 4.8 nM T64969 CP64DQ 10549169 IC50 > 5000 nM T64969 CSG53A 10549915 IC50 = 377 nM T64969 CXFB12 10555151 IC50 = 7000 nM T64969 CGAW17 10562306 IC50 > 100000 nM T64969 C6AJI9 10562777 IC50 > 100000 nM T64969 C95SZN 10564143 IC50 = 58800 nM T64969 CR91ZK 10564707 IC50 = 420 nM T64969 CW16DN 10568777 IC50 = 10 nM T64969 CX67AG 10569366 IC50 = 46 nM T64969 CE5L6D 10587839 IC50 > 100000 nM T64969 C1ICU3 10589889 IC50 = 860 nM T64969 CP8J4O 10590515 IC50 = 1270 nM T64969 CM8N6L 10593765 IC50 > 100000 nM T64969 C64CRU 10599506 IC50 > 10000 nM T64969 CF8IH9 10600888 IC50 = 3.9 nM T64969 COB2X8 10602350 IC50 = 7000 nM T64969 CY51ET 10611103 IC50 > 10000 nM T64969 CI30LZ 10613858 IC50 > 100000 nM T64969 CTG7H5 10614224 IC50 = 7830 nM T64969 C0LHE5 10615400 IC50 = 25 nM T64969 CWU4L7 10616703 IC50 = 10000 nM T64969 CNE92Q 10616753 IC50 = 230 nM T64969 CX8R0T 10618464 IC50 = 5400 nM T64969 CZ5L3U 10635276 IC50 = 200 nM T64969 CH6Z3L 10635478 IC50 > 100000 nM T64969 CB97UD 10636005 IC50 > 100000 nM T64969 C0C8QK 10638407 IC50 = 170 nM T64969 C1JY5N 10638517 IC50 = 25700 nM T64969 CG93BK 10640018 IC50 > 10000 nM T64969 C2UWA0 10658651 IC50 > 100000 nM T64969 CZ78VR 10660240 IC50 = 820 nM T64969 CZ40OF 10660724 IC50 > 5000 nM T64969 C64DFG 10662351 IC50 = 0.48 nM T64969 C5L0IX 10663368 IC50 > 100000 nM T64969 C9Z7XH 10663503 IC50 > 100000 nM T64969 C5M0HJ 10670094 IC50 = 45 nM T64969 CKA30X 10671481 IC50 = 0.51 nM T64969 CFGL61 10672994 IC50 = 6.6 nM T64969 CDV84T 10673774 IC50 = 1.8 nM T64969 CR9N8Z 10674806 IC50 > 100000 nM T64969 CH1G6P 10682457 IC50 = 44000 nM T64969 CLQP93 10683468 IC50 > 20000 nM T64969 CAVX96 10686149 IC50 > 100000 nM T64969 C51VNS 10691590 IC50 = 0.69 nM T64969 C6BK7Q 10691652 IC50 = 2.1 nM T64969 CK85TP 10692159 IC50 = 3000 nM T64969 C0AOG5 10696486 IC50 = 21 nM T64969 C7INC2 10706114 IC50 = 1250 nM T64969 CU6G5Y 10708835 IC50 > 100000 nM T64969 C54UAK 10728035 IC50 > 100000 nM T64969 CZVK65 10729749 IC50 = 550 nM T64969 CJO8Q1 10738332 IC50 = 1360 nM T64969 CN8GS6 10738988 IC50 = 1.2 nM T64969 CVX5L1 10742427 IC50 = 27 nM T64969 CXSH91 10753550 IC50 > 100000 nM T64969 C25MWP 10754509 IC50 > 10000 nM T64969 CVPW04 10755069 IC50 > 100000 nM T64969 CYAL86 10759828 IC50 = 3.3 nM T64969 CVO13S 10759989 IC50 = 41000 nM T64969 CD26KN 10760134 IC50 > 5000 nM T64969 CL0XH6 10762274 IC50 = 8000 nM T64969 CQO0A2 10762478 IC50 > 5000 nM T64969 C3WR0Q 10779668 IC50 > 100000 nM T64969 C7YJ4L 10782259 IC50 = 1.6 nM T64969 CF5T1H 10783444 IC50 = 19300 nM T64969 CFK51I 10784704 IC50 > 5000 nM T64969 C71QOK 10789593 IC50 = 1.5 nM T64969 C62FWK 10791534 IC50 = 88 nM T64969 C1OXH6 10803234 IC50 = 8 nM T64969 CT7O1G 10803426 IC50 = 10000 nM T64969 CH7Q9F 10804454 IC50 = 14000 nM T64969 C3QT8I 10806455 IC50 = 360 nM T64969 CNC84J 10811119 IC50 > 10000 nM T64969 CK0W6X 10815675 IC50 = 0.78 nM T64969 C89PRO 10826146 IC50 = 2500 nM T64969 CRJM76 10826740 IC50 = 16300 nM T64969 CDP61C 10832923 IC50 = 108 nM T64969 C3TCG9 10834960 IC50 > 5000 nM T64969 CWX4V1 10838598 IC50 = 2.7 nM T64969 CYPB29 10841700 IC50 = 6.7 ug.mL-1 T64969 C18MDA 10848423 IC50 = 570 nM T64969 C49OYX 10850623 IC50 > 10000 nM T64969 C01KXI 10854884 IC50 = 0.75 nM T64969 CGFO65 10856252 IC50 > 20000 nM T64969 C9QG7J 10868706 IC50 = 8400 nM T64969 C8IZ4B 10870494 IC50 = 24 nM T64969 CI5FC1 10875157 IC50 = 100000 nM T64969 C67ZFI 10880751 IC50 = 29 nM T64969 CTI84S 10884588 IC50 = 960 nM T64969 C7DK8H 10885120 IC50 = 2700 nM T64969 CA8J0B 10902421 IC50 = 335 nM T64969 CT7CA1 10905749 IC50 = 38 nM T64969 CJ4P5T 10905857 IC50 > 100000 nM T64969 CP5XT0 10906920 IC50 = 89.13 nM T64969 CBM57K 10918242 IC50 = 10471.29 nM T64969 CF9O7M 10926736 IC50 = 9300 nM T64969 CIRP84 10928765 IC50 = 5220 nM T64969 C60QTH 10938977 IC50 = 238 nM T64969 CI01XA 10951285 IC50 = 2640 nM T64969 CEKW21 10972694 IC50 = 560 nM T64969 C1I6VX 10973080 IC50 = 4840 nM T64969 CTY19K 10973186 IC50 = 250 nM T64969 COE13S 10983483 IC50 = 2290 nM T64969 C90YUA 10992313 IC50 = 11 nM T64969 C2AK4W 11005320 IC50 = 930 nM T64969 C3OM5X 11012217 IC50 = 13350 nM T64969 C0Y5PH 11016075 IC50 = 330 nM T64969 CM4JD2 11037303 IC50 = 7500 nM T64969 CJ05CL 11048367 IC50 > 30000 nM T64969 C9QI8E 11055442 IC50 = 8000 nM T64969 C2FPI5 11071370 IC50 = 150 nM T64969 C3UTD8 11080556 IC50 = 25 nM T64969 CR91TM 11102890 IC50 = 2880 nM T64969 C8TA4Z 11129889 IC50 > 100000 nM T64969 CR2O3F 11155047 IC50 > 10000 nM T64969 COB20T 11157041 IC50 = 768 nM T64969 CUIX38 11157794 IC50 = 30 nM T64969 C2W5OA 11165103 IC50 = 6900 nM T64969 C0VD5M 11168387 IC50 = 345 nM T64969 CSZ6B2 11168731 IC50 = 650 nM T64969 CQ7PU5 11178756 IC50 = 36 nM T64969 C7XU5W 11180271 IC50 = 24 nM T64969 C9Z6AG 11180494 IC50 = 500 nM T64969 CHV1P9 11180599 IC50 = 250 nM T64969 C2B7HJ 11180905 IC50 = 31 nM T64969 CUVW02 11186266 IC50 = 7500 nM T64969 CRG7B6 11192261 IC50 = 277 nM T64969 CA6L9Y 11192678 IC50 = 20 nM T64969 C2PMR9 11192753 IC50 = 15 nM T64969 CA07YO 11193143 IC50 = 574 nM T64969 CABZ27 11197585 IC50 = 7000 nM T64969 CQG17S 11202074 IC50 = 1020 nM T64969 C0K8NB 11202869 IC50 = 770 nM T64969 C16HXD 11203436 IC50 = 45 nM T64969 C7H8AD 11203663 IC50 = 42 nM T64969 C87QSN 11203886 IC50 = 100 nM T64969 C2NUG6 11210620 IC50 = 1000 nM T64969 C1YB7C 11220978 IC50 = 40 nM T64969 CNZ2H8 11226874 IC50 = 770 nM T64969 CMZ8S5 11227115 IC50 = 11 nM T64969 C4HUM2 11232168 IC50 = 250 nM T64969 CIJG62 11232492 IC50 = 8900 nM T64969 CH7D3X 11233762 IC50 > 100000 nM T64969 CD43EZ 11234126 IC50 = 900 nM T64969 C2W5RC 11235063 IC50 > 50000 nM T64969 C98HRX 11237508 IC50 = 185 nM T64969 CXN98V 11238293 IC50 = 341 nM T64969 CSX6P5 11238512 IC50 = 34 nM T64969 CWOU43 11238694 IC50 = 110 nM T64969 CG07FL 11238864 IC50 = 360 nM T64969 C0QN4V 11238875 IC50 = 343 nM T64969 COI7A0 11245620 IC50 = 10000 nM T64969 CU27LB 11246488 IC50 = 0.66 nM T64969 CGP6U2 11249521 IC50 = 1191 nM T64969 CO97YK 11249776 IC50 = 23 nM T64969 CJ02WR 11249881 IC50 = 223 nM T64969 CWF87N 11260603 IC50 = 372 nM T64969 CNBX16 11270660 IC50 = 2730 nM T64969 CR35NY 11273032 IC50 = 28 nM T64969 CO2E3W 11280238 IC50 > 50000 nM T64969 CUO27S 11282791 IC50 > 500 nM T64969 C5EO4X 11284905 IC50 = 34 nM T64969 CJ6R3N 11284937 IC50 = 65 nM T64969 CIV3Y6 11285080 IC50 = 282 nM T64969 C8FGR1 11288910 IC50 = 3250 nM T64969 CI63ZB 11291617 IC50 = 3400 nM T64969 CBOP58 11293798 Ki > 10000 nM T64969 C0HM3D 11293802 IC50 = 1000 nM T64969 CH02JX 11296170 IC50 = 195 nM T64969 C5Z6NC 11296256 IC50 = 163 nM T64969 CU9ER4 11296411 IC50 = 238 nM T64969 CG7VP5 11302688 IC50 = 5800 nM T64969 C84VYL 11303451 IC50 = 10 nM T64969 C6ZF7L 11303620 IC50 = 6000 nM T64969 CP3BM8 11307161 IC50 = 12700 nM T64969 C18BHK 11307255 IC50 = 445 nM T64969 C64SCF 11307581 IC50 = 32 nM T64969 C6OQC2 11307602 IC50 = 26 nM T64969 CZN3Q6 11307866 IC50 = 82 nM T64969 CANY24 11311217 IC50 = 100000 nM T64969 C0SO6D 11312797 IC50 = 412.8 nM T64969 CRD9E5 11314043 IC50 = 45000 nM T64969 CR9E2X 11316711 IC50 = 6.4 nM T64969 CLX54H 11317348 IC50 > 10000 nM T64969 CRN20W 11326156 IC50 = 37 nM T64969 C2TP7E 11327841 IC50 = 6300 nM T64969 CM48NO 11336573 IC50 = 2000 nM T64969 CKY3E2 11338122 IC50 > 50000 nM T64969 CF3W8U 11338513 IC50 = 1900 nM T64969 CSZ8P5 11340298 IC50 = 250 nM T64969 CT7CG8 11341400 IC50 = 13000 nM T64969 CXI48D 11342107 IC50 = 165 nM T64969 C8FQY5 11342284 IC50 = 31 nM T64969 CO2E6V 11342331 IC50 = 7 nM T64969 CLA1W0 11342405 IC50 = 75 nM T64969 C3KC4P 11353443 IC50 = 53 nM T64969 C49AZU 11354013 IC50 = 16 nM T64969 CDZR14 11357877 IC50 = 100 nM T64969 C0J2TB 11359024 IC50 = 50 nM T64969 C26BZX 11362471 Ki > 10000 nM T64969 CK14GM 11365122 IC50 = 111 nM T64969 C5WI2V 11365297 IC50 = 20 nM T64969 CX5FE9 11365342 IC50 = 51 nM T64969 CYF58P 11365726 IC50 = 125 nM T64969 C3OCV2 11371778 IC50 = 7100 nM T64969 C43NPS 11373886 IC50 = 30 nM T64969 CN4O0Q 11376079 IC50 = 894 nM T64969 CT3W2J 11376208 IC50 = 100 nM T64969 C4H0ZP 11380375 IC50 = 150 nM T64969 C10XFS 11382411 IC50 = 10 nM T64969 C3WYU1 11387244 IC50 = 340 nM T64969 CWXB93 11397177 Ki > 10000 nM T64969 CA9N1G 11398437 IC50 = 519 nM T64969 CN4WA3 11398461 IC50 = 130 nM T64969 CBV84Q 11398999 IC50 = 64 nM T64969 C2V7RQ 11399289 IC50 = 10 nM T64969 CY76XJ 11399310 IC50 = 214 nM T64969 C6UXH4 11399331 IC50 = 188 nM T64969 CV2IN9 11404920 IC50 = 25 nM T64969 CX25IH 11407794 IC50 = 365 nM T64969 CV5IR8 11410608 IC50 = 24 nM T64969 C9N3PO 11410634 IC50 = 400 nM T64969 CG7ES9 11410940 IC50 = 221 nM T64969 C15VAK 11420132 IC50 = 250 nM T64969 C94QJA 11420204 IC50 = 7 nM T64969 C1I4JO 11421443 IC50 = 41 nM T64969 CTCG60 11421783 IC50 = 401 nM T64969 CU6FD4 11421877 IC50 = 380 nM T64969 C0APW4 11422034 IC50 > 10000 nM T64969 C0KWX9 11422340 IC50 = 98 nM T64969 C5KWS9 11422548 IC50 = 321 nM T64969 C7AI2V 11432911 IC50 > 25000 nM T64969 C3EXM4 11440028 IC50 > 50000 nM T64969 CYD2A6 11440253 IC50 = 10 nM T64969 C3PFX4 11444623 IC50 = 78 nM T64969 CXV39N 11444862 IC50 = 362 nM T64969 CQ27HA 11452941 IC50 = 2000 nM T64969 CWI62M 11454712 IC50 = 35 nM T64969 C4LZ0F 11455794 IC50 = 285 nM T64969 CFHP63 11456360 IC50 = 990 nM T64969 C7I6AG 11474111 IC50 > 100000 nM T64969 C6M9NC 11477626 IC50 = 5500 nM T64969 CD8RQ7 11478340 IC50 = 403 nM T64969 CVFE14 11478925 IC50 = 68 nM T64969 CA0E8N 11484663 IC50 = 1100 nM T64969 C5O2TE 11486373 IC50 = 1000 nM T64969 C62KHL 11489786 IC50 = 45 nM T64969 CG7XZ1 11490270 IC50 = 63 nM T64969 CKU96Z 11490477 IC50 = 1569 nM T64969 CZI6D9 11493632 IC50 = 10000 nM T64969 C0H6QS 11495680 IC50 = 55 nM T64969 C6-AUG 11496207 IC50 = 44 nM T64969 C40GHQ 11502866 IC50 = 79 nM T64969 CIW9L5 11502867 IC50 = 10 nM T64969 CLWG73 11502887 IC50 = 74 nM T64969 C08APU 11503073 IC50 = 31 nM T64969 C2JD4P 11509595 IC50 = 10.08 nM T64969 CK2Q0X 11516978 IC50 = 120 nM T64969 CR0M9S 11517095 IC50 = 918 nM T64969 CH2IZ9 11517688 IC50 = 5200 nM T64969 CU13WV 11518389 IC50 = 0.5 nM T64969 C91JCX 11518627 IC50 = 8 nM T64969 CF0YW7 11518637 IC50 = 11 nM T64969 CV3NK7 11524106 IC50 = 4.5 nM T64969 CQ63ER 11524582 IC50 = 31.62 nM T64969 C5V7WY 11525136 IC50 = 21700 nM T64969 CI5ET2 11525434 IC50 = 21 nM T64969 CPE53F 11526238 IC50 = 6 nM T64969 C7HMO6 11526786 IC50 > 10000 nM T64969 CL7X4Q 11530963 IC50 = 32000 nM T64969 C5BM4T 11531799 IC50 = 9 nM T64969 C53OSD 11532048 IC50 = 40 nM T64969 CT75DZ 11532242 IC50 = 4.5 nM T64969 CC4QM5 11532676 IC50 = 20 nM T64969 CY6L8I 11532718 IC50 > 10000 nM T64969 C1SGF3 11533556 IC50 = 14 nM T64969 CSKF56 11538667 IC50 = 19.1 nM T64969 CTG83F 11539329 Ki > 1800 nM T64969 C5VO2C 11539461 IC50 = 3.1 nM T64969 C4SNI6 11542889 IC50 > 10000 nM T64969 CGN83M 11544306 IC50 = 10000 nM T64969 C01FVM 11546457 IC50 = 20 nM T64969 CLBH14 11547991 IC50 = 9 nM T64969 C37WYM 11552033 IC50 = 10.9 nM T64969 C7WO0I 11552307 IC50 = 16 nM T64969 C23INE 11552309 IC50 = 9.31 nM T64969 CX6KD1 11553647 IC50 = 6.8 nM T64969 CPT4K5 11554463 IC50 = 294 nM T64969 C3MD0B 11557040 IC50 = 5 nM T64969 CI50OC 11558284 IC50 = 4 nM T64969 C2DM7W 11560794 IC50 = 19300 nM T64969 CB46CA 11561058 IC50 = 77 nM T64969 CS2U5G 11561468 IC50 = 33 nM T64969 CZ9N6O 11561637 IC50 = 30700 nM T64969 CXT51U 11561779 IC50 = 8 nM T64969 CACS26 11561968 Ki > 2000 nM T64969 CNBM81 11562171 IC50 = 9 nM T64969 CKUR82 11568720 IC50 = 1.3 nM T64969 CNV08X 11569158 IC50 = 22 nM T64969 CZ1H0X 11569258 IC50 = 2800 nM T64969 C2R0XV 11569434 IC50 = 104 nM T64969 CO8UB2 11569903 IC50 = 327 nM T64969 COGM15 11574917 IC50 = 1000 nM T64969 CI4P0T 11575228 IC50 = 27000 nM T64969 CU3Q1T 11576231 IC50 = 40 nM T64969 CA74QZ 11581908 IC50 = 5010 nM T64969 CM8NI3 11582856 IC50 = 45900 nM T64969 CW5ZP3 11583431 IC50 > 100000 nM T64969 CO9KP5 11583459 IC50 = 9600 nM T64969 CXMY21 11583563 IC50 = 76 nM T64969 C8ZHL0 11589515 IC50 = 67 nM T64969 C8E5DA 11589674 IC50 > 10000 nM T64969 CMIL86 11590363 Ki > 1800 nM T64969 CN31OR 11590557 IC50 = 1.7 nM T64969 CCPK51 11590799 IC50 = 32 nM T64969 CK4E6V 11591222 IC50 = 2000 nM T64969 CR06MA 11595844 IC50 = 1.4 nM T64969 CE6P8L 11595868 IC50 = 10000 nM T64969 C0NV9Y 11596881 IC50 = 8 nM T64969 CHZ38O 11597061 IC50 = 17 nM T64969 CP1O4N 11597180 IC50 = 17 nM T64969 CR1FG0 11604864 IC50 = 4.3 nM T64969 CC48BK 11605761 IC50 = 60 nM T64969 CFEK68 11606101 IC50 = 3 nM T64969 CF7P3R 11611500 IC50 = 18 nM T64969 C85QTY 11611655 IC50 = 1500 nM T64969 C7TA0C 11612021 IC50 = 42 nM T64969 C9T3VC 11613187 IC50 = 2.7 nM T64969 CSKW87 11617204 IC50 = 240 nM T64969 CEO7I2 11618876 IC50 = 8.95 nM T64969 CZJU74 11619195 IC50 = 5900 nM T64969 C7SFP9 11619763 IC50 = 333 nM T64969 CO68CD 11619972 IC50 = 1 nM T64969 C1BLZ5 11620055 IC50 = 9 nM T64969 C5B3XJ 11620410 IC50 > 25000 nM T64969 CJ6NA8 11620487 IC50 < 1 nM T64969 C5KHN0 11625514 IC50 = 50 nM T64969 C9ZD2E 11626406 IC50 = 1029 nM T64969 CSM62L 11626920 IC50 > 30000 nM T64969 CGX96V 11626927 IC50 < 10000 nM T64969 C1VOW6 11627264 IC50 = 91 nM T64969 CQK9C3 11627337 IC50 < 1 nM T64969 C65ZXO 11632139 IC50 = 10000 nM T64969 CG0K4A 11632391 IC50 = 1.7 nM T64969 CK34LS 11632737 IC50 > 50000 nM T64969 CR1GI3 11633096 IC50 = 9 nM T64969 CB4YR6 11634425 IC50 = 17 nM T64969 C19LFT 11634645 IC50 = 5 nM T64969 CFM2Y4 11640405 IC50 > 10000 nM T64969 C3DIA4 11640601 IC50 > 100000 nM T64969 CW5A2S 11640889 IC50 = 32 nM T64969 C9T6SC 11640926 Ki > 1800 nM T64969 CE5MY2 11645981 IC50 = 10000 nM T64969 C9SPF4 11654839 IC50 = 340 nM T64969 C63JRY 11655241 IC50 = 1200 nM T64969 CA8X1L 11655791 IC50 = 0.64 nM T64969 C1AX2K 11656050 IC50 = 12 nM T64969 C79EDK 11657332 IC50 = 15 nM T64969 COI6C7 11660896 IC50 = 0.38 nM T64969 C24GRQ 11661959 IC50 = 20 nM T64969 C59AXH 11663284 IC50 = 16 nM T64969 CP04JC 11666231 IC50 > 10000 nM T64969 C8BLT1 11667173 IC50 = 32.2 nM T64969 CK64UO 11668874 IC50 = 2900 nM T64969 C1ZAE8 11669455 IC50 = 30 nM T64969 C5QM4L 11670167 IC50 = 1430 nM T64969 C9YK5E 11675213 IC50 = 22 nM T64969 CVLA25 11675714 IC50 = 500 nM T64969 CDA46H 11675978 IC50 = 16 nM T64969 C75CNZ 11678194 IC50 = 6.7 nM T64969 C0YOG3 11681189 IC50 = 199.53 nM T64969 C7T9ES 11681588 IC50 = 150 nM T64969 CS72ED 11682843 IC50 = 20 nM T64969 CQ69CR 11683171 IC50 = 204 nM T64969 C9YA5W 11683816 IC50 = 47 nM T64969 CJ9KN7 11683817 IC50 > 10000 nM T64969 C6GQ3R 11684059 IC50 = 1600 nM T64969 CQA9W7 11684098 IC50 = 150 nM T64969 C1P8JC 11684684 IC50 = 7 nM T64969 CP3U0W 11684933 IC50 = 397 nM T64969 C8AEX7 11687971 IC50 > 200000 nM T64969 C0UGQ3 11689490 IC50 = 10000 nM T64969 CU0E8O 11690457 Ki > 10000 nM T64969 C5JNW3 11690494 IC50 > 100000 nM T64969 C7I9FP 11690513 IC50 = 700 nM T64969 CLC53E 11691173 IC50 = 10 nM T64969 CP8WJ3 11691483 IC50 > 10000 nM T64969 C6QI9A 11698674 IC50 = 38 nM T64969 CKF8X5 11698913 IC50 = 13 nM T64969 C5J8NA 11703562 IC50 = 17 nM T64969 CX6IC8 11705545 IC50 > 100000 nM T64969 CB0AP2 11705863 Ki > 10000 nM T64969 CI7O1T 11706282 IC50 = 97 nM T64969 C1XNT2 11710303 IC50 = 99 nM T64969 CXOF82 11711590 IC50 = 15 nM T64969 CLY3T0 11712237 IC50 = 1100 nM T64969 CWX07A 11712609 IC50 = 216 nM T64969 C93EKF 11712721 IC50 = 70 nM T64969 CXKT32 11712931 IC50 = 1.66 nM T64969 C4YWU2 11713043 IC50 = 4.5 nM T64969 CR51YI 11717370 IC50 = 676 nM T64969 C1FTX3 11719305 IC50 = 35 nM T64969 CZY05V 11719421 IC50 = 965 nM T64969 C8WQ9F 11719423 IC50 = 4.2 nM T64969 CC3XP1 11720499 IC50 = 23 nM T64969 C8QI0K 11723086 IC50 > 20000 nM T64969 CFJ4I7 11723151 IC50 > 100000 nM T64969 C45EWD 11723489 IC50 > 7000 nM T64969 C9HC4M 11726643 IC50 = 3900 nM T64969 C9P0VD 11729539 IC50 > 100000 nM T64969 CQ3R5E 11733863 IC50 = 130 nM T64969 C7C2FM 11737638 IC50 > 100000 nM T64969 CPY1Z2 11740563 IC50 = 800 nM T64969 CP7AH3 11755812 IC50 = 50000 nM T64969 CWL34S 11756855 IC50 > 100000 nM T64969 C43NTX 11762902 IC50 = 550 nM T64969 C3J7MT 11777791 IC50 > 100000 nM T64969 CGYV23 11779501 IC50 = 360 nM T64969 C9Z7WU 11779874 IC50 > 20000 nM T64969 CV2RD0 11786660 IC50 = 140 nM T64969 CTZ60E 11786930 IC50 = 32 nM T64969 CF2M6O 11797642 IC50 > 20000 nM T64969 CJPT37 11799155 IC50 = 1.5 nM T64969 CH37DA 11802348 IC50 = 3000 nM T64969 C4Q1AE 11817879 IC50 = 110 nM T64969 CYO7K5 11822927 IC50 = 482 nM T64969 C9JT4S 11847343 IC50 > 10000 nM T64969 CHR92S 11858109 IC50 = 1700 nM T64969 CQF23E 11952856 IC50 < 10 nM T64969 C0A4TX 11955109 IC50 = 3 nM T64969 CESM43 11955112 IC50 = 9 nM T64969 CAGY67 11955434 IC50 = 13 nM T64969 CM50UH 12000646 IC50 > 10000 nM T64969 CKPW61 12211388 IC50 = 2710 nM T64969 C2Y5BU 12213273 IC50 = 10 nM T64969 CD6KA7 12241082 IC50 = 2 ug.mL-1 T64969 CJ5K4M 12341776 IC50 = 52 nM T64969 C78FCI 12482705 IC50 = 20040 nM T64969 C9MHX7 12484326 IC50 > 100000 nM T64969 C6PYI9 12814948 IC50 = 75000 nM T64969 C40ZMY 13038269 IC50 = 156 nM T64969 C0NBY4 13041145 IC50 = 1080 nM T64969 CT0R3M 13126887 IC50 = 30 nM T64969 CWUK08 13492269 IC50 = 1900 nM T64969 CO74KJ 13492270 IC50 = 2100 nM T64969 C9J0ID 13492273 IC50 = 77500 nM T64969 CHD0C6 13492275 IC50 = 75100 nM T64969 CR1H5O 13492276 IC50 > 50000 nM T64969 C7LN2W 13492279 IC50 = 560 nM T64969 CJXA95 13492280 IC50 = 1900 nM T64969 C2QEX8 13492281 IC50 = 3000 nM T64969 CC16HJ 13492282 IC50 = 110 nM T64969 CE0IS9 13492283 IC50 > 100000 nM T64969 CC70UD 13498036 IC50 > 100000 nM T64969 CG0VW8 13965155 IC50 = 17190 nM T64969 C5MI4N 14246200 IC50 = 60 nM T64969 CXPU45 14246203 IC50 = 110 nM T64969 C52VQJ 14459363 IC50 = 20 ug.mL-1 T64969 CY1I9N 14459364 IC50 = 2 ug.mL-1 T64969 C2HK6N 14459365 IC50 = 5 ug.mL-1 T64969 CRB23M 14489592 IC50 = 412.3 nM T64969 CQA20E 14547432 IC50 = 20000 nM T64969 C2Z8DQ 14624081 IC50 = 4600 nM T64969 C05MWB 14738184 IC50 = 31768.74 nM T64969 CY6H5R 14758720 IC50 = 56.48 nM T64969 CQ2MO7 14800296 IC50 > 6 ug.mL-1 T64969 CJ1XI6 14800297 IC50 > 6 ug.mL-1 T64969 CCG0R9 14862523 IC50 = 2800 nM T64969 C9EOJ3 14862524 IC50 = 50 nM T64969 CZ4C8O 14862525 IC50 = 300 nM T64969 C8ID0S 14862526 IC50 = 2500 nM T64969 C8AF0C 14862527 IC50 = 1500 nM T64969 CMIY48 14862528 IC50 = 1800 nM T64969 CLQJ06 14862530 IC50 = 600 nM T64969 CO1WA7 14862532 IC50 = 500 nM T64969 C4P3OG 14862533 IC50 = 400 nM T64969 CICQ96 14862534 IC50 = 4000 nM T64969 C3HEO0 14862536 IC50 = 1300 nM T64969 CAJ79W 14862537 IC50 = 4800 nM T64969 CAY7Z2 14862538 IC50 > 100000 nM T64969 CI5KD3 14862539 IC50 = 1000 nM T64969 CTM1N7 14862540 IC50 = 5000 nM T64969 CK60ZN 14862550 IC50 > 50000 nM T64969 CHC25I 14862551 IC50 = 20000 nM T64969 CUMI23 14943555 IC50 = 15000 nM T64969 CRZG26 14943556 IC50 = 6100 nM T64969 C5M6ZT 14943557 IC50 = 28700 nM T64969 CJ5RZ6 14994201 IC50 = 400 nM T64969 CW48TD 15159374 IC50 = 689 nM T64969 CK8XF4 15209376 IC50 = 1500 nM T64969 CPK05U 15249955 IC50 = 100000 nM T64969 CDGF78 15282555 IC50 = 1300 nM T64969 CVU54Q 15324448 IC50 = 19730 nM T64969 CIL1R3 15411595 IC50 = 160000 nM T64969 CKU75C 15520888 IC50 = 1643.6 nM T64969 CQ9Z0L 15550318 IC50 = 5100 nM T64969 CW4R6I 15550657 IC50 = 374.8 nM T64969 CJ81ZO 15550658 IC50 = 6266.2 nM T64969 CN2Z1V 15598735 IC50 = 10 ug.mL-1 T64969 CL81NH 15598736 IC50 = 10 ug.mL-1 T64969 C01JGR 15598739 IC50 = 5 ug.mL-1 T64969 CR7SM0 15598740 IC50 = 4 ug.mL-1 T64969 CSFP09 15598743 IC50 = 2 ug.mL-1 T64969 CAG6P9 15598744 IC50 = 10 ug.mL-1 T64969 C6JS5O 15603105 IC50 = 5.35 nM T64969 CP8OW6 15858662 IC50 = 500 nM T64969 CUI6E5 15858664 IC50 = 170 nM T64969 C6PZU3 15858665 IC50 = 350 nM T64969 CEMH32 15858666 IC50 = 1530 nM T64969 CK5QI3 15858667 IC50 = 1120 nM T64969 CFHW20 15942947 IC50 = 85600 nM T64969 C1O8MK 15946672 IC50 = 9 nM T64969 C7LB4I 15949613 IC50 > 10000 nM T64969 C21YPU 16004616 IC50 = 90400 nM T64969 CFPW41 16007116 Ki > 1800 nM T64969 CS28LD 16035342 IC50 = 40 nM T64969 C5KS0Q 16036986 IC50 = 10 nM T64969 CQM4R7 16036987 IC50 = 15 nM T64969 CBU5P8 16037083 IC50 = 12 nM T64969 C69NIP 16037084 IC50 = 13 nM T64969 CM8IN2 16037085 IC50 = 4 nM T64969 C91PSH 16037086 IC50 = 12 nM T64969 CDZR21 16037089 IC50 = 25 nM T64969 CZ0UJ7 16037184 IC50 = 43 nM T64969 CAZ34B 16037276 IC50 = 3300 nM T64969 C1DO0X 16037278 IC50 = 187 nM T64969 CQR5O7 16042971 IC50 = 1500 nM T64969 CZK8V6 16043304 IC50 > 10000 nM T64969 CH9LO8 16044634 IC50 = 7700 nM T64969 C3ZC6E 16045442 IC50 < 1 nM T64969 C2MH6N 16045730 IC50 = 1 nM T64969 CD2F8V 16046116 IC50 = 690 nM T64969 CQW10N 16066845 IC50 = 30 nM T64969 C3GW0S 16069809 IC50 = 83900 nM T64969 CQG45C 16109001 IC50 = 25000 nM T64969 CZC0H1 16116961 IC50 = 180 nM T64969 C6D8MB 16118310 Ki = 1.6 nM T64969 CL5IF2 16214946 IC50 > 30000 nM T64969 CY1CB3 16215851 IC50 = 60 nM T64969 CXUO14 16457485 IC50 = 311 nM T64969 CVCD64 16663769 IC50 = 0.1 nM T64969 CU56EW 16664858 IC50 > 10000 nM T64969 C2IF3P 16678352 IC50 = 3580 nM T64969 C3IO1C 16679060 IC50 > 10000 nM T64969 C5WIS9 16719846 IC50 = 71 nM T64969 CCD20J 16719847 IC50 = 2200 nM T64969 CT68JW 16719965 IC50 = 970 nM T64969 C02KXR 16719966 IC50 = 4.4 nM T64969 CMLX63 16719967 IC50 = 3960 nM T64969 CHZ20P 16730263 IC50 = 20 nM T64969 C1Y2JH 16745310 IC50 = 799.3 nM T64969 CN8WX3 16757526 IC50 = 22000 nM T64969 CEXL56 17271861 IC50 = 13230 nM T64969 CQY57T 17747104 IC50 = 70 nM T64969 C4BQ6L 17747105 IC50 = 8 nM T64969 CKU29X 17747134 IC50 = 12 nM T64969 C5YZ9V 17747138 IC50 = 16 nM T64969 C95LWR 17747139 IC50 = 5 nM T64969 CW61OK 17747208 IC50 = 32 nM T64969 CQ7RH3 17747242 IC50 = 13 nM T64969 CXD23O 17747243 IC50 = 24 nM T64969 C2VL8S 17747279 IC50 = 47 nM T64969 C8AM0W 17747280 IC50 = 23 nM T64969 CEG7O8 17747281 IC50 = 14 nM T64969 CR4PF2 17747282 IC50 = 44 nM T64969 CYB3N5 17747309 IC50 = 20 nM T64969 CC2W0F 17747311 IC50 = 23 nM T64969 CS9O2H 17747339 IC50 = 48 nM T64969 CL83TA 17747341 IC50 = 104 nM T64969 C1VC9E 17747343 IC50 = 14 nM T64969 C7Q0ZD 17747376 IC50 = 57 nM T64969 CUT1G2 17747492 IC50 = 33 nM T64969 CNRV46 17747535 IC50 = 27 nM T64969 CL9BQ6 17748275 IC50 = 25000 nM T64969 CAV9R6 17757434 IC50 > 20000 nM T64969 C8AH1I 17758019 IC50 = 1000 nM T64969 C1GKL6 17758020 IC50 > 5000 nM T64969 CO6LR5 17758240 IC50 = 500 nM T64969 CU0MF7 17758241 IC50 = 3300 nM T64969 CE73IF 17758353 IC50 = 5000 nM T64969 CH9TR6 17758354 IC50 = 156 nM T64969 CA79FH 17758358 IC50 > 5000 nM T64969 CSA23C 17759556 IC50 > 20000 nM T64969 C56YOG 17759673 IC50 = 2080 nM T64969 CIL8G9 17759675 IC50 > 20000 nM T64969 C57NRL 17759787 IC50 = 2900 nM T64969 C3D7WE 17874201 IC50 > 200000 nM T64969 C35IWY 17938625 IC50 = 4000 nM T64969 C7ZK1E 17938633 IC50 = 30000 nM T64969 CQ35AK 17953498 IC50 = 730 nM T64969 CM2HS9 18176200 IC50 = 0.6 nM T64969 C60VEN 18176234 IC50 = 0.69 nM T64969 CYD95N 18184369 IC50 = 132 nM T64969 C8NCX0 18184376 IC50 = 2110 nM T64969 C1SQC4 18184420 IC50 = 72 nM T64969 CQA78V 18382736 IC50 = 5 nM T64969 C2EBQ5 18382775 IC50 = 4 nM T64969 CZB5L4 18382784 IC50 = 100 nM T64969 C1LUP2 18382794 IC50 = 3 nM T64969 C8KJ4R 18382823 IC50 > 1000 nM T64969 CZC98J 18382853 IC50 = 1 nM T64969 C5QV1L 18382857 IC50 = 1600 nM T64969 C84KLY 18382861 IC50 = 30 nM T64969 CSPD61 18382868 IC50 = 140 nM T64969 CG4BK9 18382875 IC50 = 3 nM T64969 C8BK3Q 18382898 IC50 = 4 nM T64969 CX7F1I 18382902 IC50 = 2 nM T64969 CNE4R0 18382910 IC50 = 1 nM T64969 CML03B 18382946 IC50 = 5 nM T64969 CGXU47 18382956 IC50 = 600 nM T64969 C5BGJ8 18382993 IC50 = 2 nM T64969 CVFU60 18383007 IC50 = 9 nM T64969 CZ90LJ 18383038 IC50 = 9 nM T64969 C2R0KU 18383095 IC50 = 94 nM T64969 CBF6H0 18383099 IC50 = 500 nM T64969 C7SQ3Z 18383101 IC50 = 657 nM T64969 CQ7V2F 18383102 IC50 = 250 nM T64969 CT7GK6 18548938 IC50 > 10000 nM T64969 CX69ZL 18548951 IC50 > 10000 nM T64969 C8MQ2N 18770775 IC50 = 5500 nM T64969 CY97MC 18770784 IC50 = 100 nM T64969 CHDY96 18770788 IC50 = 600 nM T64969 C1HCE3 18770799 IC50 = 3000 nM T64969 C72EWO 18770811 IC50 = 6500 nM T64969 C4BTV7 18770818 IC50 = 3000 nM T64969 C3JP7K 18770822 IC50 > 20000 nM T64969 C1GAJ2 18770840 IC50 = 500 nM T64969 C1C0EJ 18792861 IC50 = 2540 nM T64969 C6HK0S 18792868 IC50 = 500 nM T64969 C90EQY 18792940 IC50 = 2670 nM T64969 C9PS7R 18792941 IC50 = 900 nM T64969 CIH2K0 18792942 IC50 = 400 nM T64969 CILQ48 18792962 IC50 = 13400 nM T64969 C7R5VZ 18967573 IC50 = 59 nM T64969 C3AZJ2 19037238 IC50 > 200000 nM T64969 CC7U2Q 19077486 IC50 = 79 nM T64969 CXB56W 19077488 IC50 = 57 nM T64969 C96VSF 19077498 IC50 = 49 nM T64969 CNC8P2 19077501 IC50 = 7 nM T64969 C54VNA 19077504 IC50 = 61 nM T64969 C3O9AD 19077506 IC50 = 60.2 nM T64969 CEO7V9 19077507 IC50 = 98 nM T64969 CAUO09 19077508 IC50 = 10 nM T64969 CMI72S 19077513 IC50 = 93 nM T64969 CU4R5O 19077515 IC50 = 18.1 nM T64969 CB32XU 19077516 IC50 = 71 nM T64969 CBUP69 19077520 IC50 = 87 nM T64969 C0FL3G 19888887 IC50 > 30 ug.mL-1 T64969 C0WEX3 19966997 IC50 > 100000 nM T64969 C0E2OG 20579089 IC50 > 10000 nM T64969 C3AI0N 20817111 IC50 = 2300 nM T64969 CFI0B9 21010047 IC50 = 2.61 nM T64969 C81ALS 21080010 IC50 = 0.11 nM T64969 C51HNQ 21080015 IC50 = 0.94 nM T64969 CL81VC 21100709 IC50 = 100000 nM T64969 C3EHM4 21197160 IC50 = 90000 nM T64969 CEBF05 21697320 IC50 = 150 nM T64969 CVI49J 21701562 IC50 = 5700 nM T64969 CFN6G4 21701597 IC50 = 100 nM T64969 C5B7WP 21874200 IC50 = 9 nM T64969 CBN19I 21874228 IC50 = 130 nM T64969 CLD73T 21874248 IC50 = 32 nM T64969 CYSR48 21874287 IC50 = 20 nM T64969 CWY6T7 21874402 IC50 = 660 nM T64969 C5IBJ0 21874410 IC50 = 6 nM T64969 CM3XF9 21874431 IC50 = 50 nM T64969 CRB1V5 21945809 IC50 = 490 nM T64969 CT9LP3 21945841 IC50 = 200 nM T64969 C5GIE9 21945968 IC50 = 40 nM T64969 CHU2Z3 21951965 IC50 = 80 nM T64969 CLN2G9 21952043 IC50 = 25 nM T64969 CH27DF 21988185 IC50 > 10000 nM T64969 COH4Y2 21988214 IC50 > 10000 nM T64969 CXJI39 22022153 IC50 = 100 nM T64969 CFG57O 22024915 IC50 = 2 nM T64969 C5MEX2 22024916 IC50 = 150 nM T64969 CQEN87 22055240 IC50 = 85 nM T64969 C8J9GH 22055262 IC50 = 48 nM T64969 C2RY4D 22055269 IC50 = 250 nM T64969 CPV5Z0 22132688 IC50 > 10000 nM T64969 CH5V2Q 22390479 IC50 = 210 nM T64969 C1IU0K 22390480 IC50 = 710 nM T64969 C50SLD 22390490 IC50 = 620 nM T64969 C7GK1A 22390495 IC50 = 110 nM T64969 CKV0J5 22390502 IC50 = 500 nM T64969 C5NVM0 22390522 IC50 = 220 nM T64969 C9G5RQ 22390524 IC50 = 50 nM T64969 CHF3A0 22390530 IC50 = 100 nM T64969 CD5GI0 22390536 IC50 = 110 nM T64969 C18CUK 22390541 IC50 = 200 nM T64969 C3H4NO 22390542 IC50 = 120 nM T64969 CNMZ85 22390556 IC50 = 380 nM T64969 C1CJS9 22466664 IC50 = 330.2 nM T64969 CWL0O9 22466767 IC50 = 1040 nM T64969 CF6LA9 22478260 IC50 = 90 nM T64969 CMRO51 22478297 IC50 = 80 nM T64969 C7TK3G 22478429 IC50 = 126.9 nM T64969 C2P1DL 22667101 IC50 > 10000 nM T64969 CK35BP 22667145 IC50 > 10000 nM T64969 C1PR6W 22692676 IC50 > 50000 nM T64969 CSB1G3 22692751 IC50 = 900 nM T64969 CYN49O 22692759 IC50 = 37600 nM T64969 CZRM03 22692773 IC50 = 36000 nM T64969 CB1V6E 22692848 IC50 = 2370 nM T64969 CO2R3S 22692946 IC50 = 4300 nM T64969 C9WHT0 22692968 IC50 > 100000 nM T64969 CKB7C2 22693031 IC50 > 100000 nM T64969 C6CHV3 22693234 IC50 = 9700 nM T64969 CC1U4X 22732253 IC50 = 5600 nM T64969 COB60M 23133320 IC50 = 100 nM T64969 C9QLP0 23133323 IC50 = 170 nM T64969 C4E1SO 23290441 IC50 = 0.208 nM T64969 CQMH63 23366746 IC50 = 1800 nM T64969 C6JV7W 23400934 IC50 > 7000 nM T64969 CD5S7O 23401001 IC50 > 7000 nM T64969 CV8P7G 23546054 IC50 > 40000 nM T64969 C9PF3L 23546055 IC50 = 5400 nM T64969 C2XRV0 23546056 IC50 = 1000 nM T64969 CWU9P6 23589545 IC50 = 120 nM T64969 CEN3B8 23589555 IC50 = 950 nM T64969 CRX0Q6 23625758 IC50 > 100000 nM T64969 C19TLD 23644675 IC50 = 1600 nM T64969 CX32IF 23646535 IC50 = 90 nM T64969 C4Z5YE 23646536 IC50 = 60 nM T64969 CZ6E5P 23646537 IC50 = 50 nM T64969 CG7F1M 23646539 IC50 = 610 nM T64969 C9ZSO0 23646540 IC50 = 120 nM T64969 C06CVI 23646541 IC50 = 200 nM T64969 C42ONU 23646542 IC50 = 200 nM T64969 C3T8FB 23646543 IC50 > 25000 nM T64969 CVK4Z2 23646544 IC50 = 120 nM T64969 CS31HG 23646545 IC50 = 70 nM T64969 CRQK51 23646546 IC50 = 210 nM T64969 C7O2QA 23646547 IC50 = 7400 nM T64969 C82MEJ 23646548 IC50 = 950 nM T64969 C08NIK 23646549 IC50 = 1100 nM T64969 CV75ZR 23646550 IC50 = 170 nM T64969 C2S5ZM 23661662 Ki = 3 nM T64969 CYWG82 23729145 IC50 = 490 nM T64969 COV2N4 24179332 IC50 = 10340 nM T64969 CUGY24 24202429 IC50 = 1900 nM T64969 CNWM52 24322804 IC50 = 7440 nM T64969 CLIV79 24737855 IC50 < 15 nM T64969 CH53CN 24738004 IC50 = 5.06 nM T64969 CA3I4T 24753787 IC50 > 50000 nM T64969 C7YG1N 24759534 IC50 = 1100 nM T64969 CAJ4T2 24762205 IC50 > 10000 nM T64969 CCPS81 24764502 IC50 > 35000 nM T64969 C78RNQ 24766872 IC50 = 197 ug.mL-1 T64969 CQ8SY7 24766873 IC50 > 200 ug.mL-1 T64969 C31EHS 24767187 IC50 > 20000 nM T64969 CJUK39 24770517 IC50 > 10000 nM T64969 C0EKO5 24772654 IC50 = 3300 nM T64969 CC1L8F 24777233 IC50 = 76 nM T64969 CXS1U4 24779710 IC50 = 14.1 nM T64969 C1CGU3 24782374 IC50 = 5000 nM T64969 C7DR5J 24782621 IC50 = 257 nM T64969 CFN39G 24782622 IC50 = 980 nM T64969 CE2Q3V 24786207 IC50 = 1160 nM T64969 C9PA0M 24807809 IC50 > 10000 nM T64969 CY8X0J 24811794 Ki > 10000 nM T64969 C7UPH2 24824775 IC50 = 4720 nM T64969 C61KPI 24856363 IC50 > 25000 nM T64969 C3S5KC 24863865 IC50 = 209 nM T64969 CFK2B9 24882503 IC50 = 380 nM T64969 C43HWQ 24883287 IC50 = 24 nM T64969 C8DA5Q 24883334 IC50 = 9 nM T64969 C4V9GH 24894117 IC50 = 23000 nM T64969 CZ6KD4 24894886 IC50 = 22000 nM T64969 CB5TP8 24894992 IC50 = 9000 nM T64969 C32SUJ 24894993 IC50 = 14000 nM T64969 CY8L7E 24896769 IC50 > 10000 nM T64969 CZ67RA 24897043 IC50 = 8 nM T64969 CVF5W2 24897276 IC50 = 30 nM T64969 CB2EX1 24897277 IC50 = 16 nM T64969 CN9T1Z 24897278 IC50 = 16 nM T64969 C6JA7L 24897279 IC50 = 31 nM T64969 CA5XT2 24897280 IC50 = 26 nM T64969 CN13JF 24899915 IC50 = 4.2 ug.mL-1 T64969 CBWR97 24899916 IC50 = 1.1 ug.mL-1 T64969 C9F2JD 24899917 IC50 > 10 ug.mL-1 T64969 C64MTI 24900160 IC50 = 4.2 ug.mL-1 T64969 CO2I6Q 24900161 IC50 = 6.5 ug.mL-1 T64969 CB79YC 24905143 IC50 = 954 nM T64969 C2DC9J 24905144 IC50 = 388 nM T64969 CN6V8Z 24905145 IC50 = 550 nM T64969 CSB7P5 24905148 IC50 = 12000 nM T64969 CGSF21 24905149 IC50 > 50000 nM T64969 CVDG02 24905150 IC50 = 170 nM T64969 CWH6C5 24905152 IC50 = 610 nM T64969 C0HE2Q 24905153 IC50 = 2300 nM T64969 C7QSC9 24905154 IC50 = 579 nM T64969 CO9D0K 24905155 IC50 = 12000 nM T64969 C5W9UR 24905157 IC50 = 9900 nM T64969 CC1DA3 24905158 IC50 = 5960 nM T64969 COW79F 24905159 IC50 = 100000 nM T64969 CFPA53 24905160 IC50 = 100000 nM T64969 C2O0JX 24905161 IC50 = 12800 nM T64969 CA72BE 24905162 IC50 = 100000 nM T64969 CQN6X9 24905163 IC50 = 100000 nM T64969 CD4O1F 24905165 IC50 = 8300 nM T64969 CKL48T 24905166 IC50 = 13000 nM T64969 C76VYL 24905167 IC50 = 17000 nM T64969 C7K5PU 24905168 IC50 = 4300 nM T64969 CZ57ID 24905169 IC50 = 1400 nM T64969 C2DHX9 24905170 IC50 = 100000 nM T64969 CSB96E 24905171 IC50 = 100000 nM T64969 CWZ0R2 24905172 IC50 = 15000 nM T64969 CY3B6M 24905175 IC50 = 3860 nM T64969 CW7UA3 24905176 IC50 = 10200 nM T64969 CW1V0H 24905177 IC50 = 5140 nM T64969 CO6Y0L 24905178 IC50 = 3660 nM T64969 C60NQW 24905179 IC50 = 100000 nM T64969 C4MO8B 24905180 IC50 = 3720 nM T64969 COJI47 24905181 IC50 = 1770 nM T64969 CS0B2C 24905182 IC50 = 751 nM T64969 C1H4BT 24905183 IC50 = 84 nM T64969 C4WHK9 24905184 IC50 = 11000 nM T64969 C7Q4MZ 24905185 IC50 = 179 nM T64969 CS4IP1 24905186 IC50 = 249 nM T64969 C69QWO 24905187 IC50 = 391 nM T64969 C85ANB 24905188 IC50 = 176 nM T64969 CNHD75 24905189 IC50 = 3300 nM T64969 C9JUO2 24905190 IC50 = 4600 nM T64969 CPR03K 24905191 IC50 = 1400 nM T64969 CTAG19 24905193 IC50 = 734 nM T64969 C7VJM5 24905194 IC50 = 5000 nM T64969 CEP1L3 24905195 IC50 = 964 nM T64969 CP68ZD 24905196 IC50 = 575 nM T64969 C8Z0RJ 24905197 IC50 = 768 nM T64969 CN9RT0 24905198 IC50 = 5320 nM T64969 CHI78P 24905200 IC50 = 1000 nM T64969 CO6PE8 24905201 IC50 = 220 nM T64969 CZ63HS 24905202 IC50 = 380 nM T64969 C2X0FC 24905203 IC50 = 2500 nM T64969 C0WCE3 24905204 IC50 = 34000 nM T64969 CNK50B 24905205 IC50 = 2100 nM T64969 C12DPB 24905206 IC50 = 760 nM T64969 C8N0RH 24905207 IC50 = 21000 nM T64969 CYA5G2 24905208 IC50 = 100000 nM T64969 CDV2B4 24905209 IC50 = 2900 nM T64969 CEFK68 24905210 IC50 = 15000 nM T64969 CUFP12 24905211 IC50 = 540 nM T64969 C0JG8L 24905212 IC50 = 85 nM T64969 CQ13ZI 24905215 IC50 = 25000 nM T64969 C6VI8F 24905216 IC50 = 100000 nM T64969 CXNH25 24905217 IC50 = 100000 nM T64969 C2PN9S 24905218 IC50 = 18000 nM T64969 C9O2AL 24905219 IC50 = 18000 nM T64969 CIT7U8 24905220 IC50 = 100000 nM T64969 CMD26S 24905221 IC50 = 955 nM T64969 C4R8WC 24905222 IC50 = 539 nM T64969 C47SHA 24905223 IC50 = 1100 nM T64969 C1DY2R 24905224 IC50 = 571 nM T64969 CS0XF9 24905225 IC50 = 70000 nM T64969 CG5VX2 24905226 IC50 = 6700 nM T64969 C57QEO 24905227 IC50 = 1400 nM T64969 C7CG5E 24905228 IC50 = 7000 nM T64969 CHP5D1 24905229 IC50 = 29000 nM T64969 CXP09S 24905230 IC50 = 100000 nM T64969 CY7XG1 24905231 IC50 = 100000 nM T64969 C7JFQ2 24905232 IC50 = 12000 nM T64969 C2JM1P 24905233 IC50 = 100000 nM T64969 CC3BF0 24905234 IC50 = 10000 nM T64969 CE57FI 24905235 IC50 = 10000 nM T64969 CUP20O 24905236 IC50 = 100000 nM T64969 CLC6Q2 24905237 IC50 = 8900 nM T64969 C9M1GI 24905238 IC50 = 9000 nM T64969 CVD72F 24905239 IC50 = 207 nM T64969 CK38IZ 24905240 IC50 = 2600 nM T64969 CO2V5E 24905241 IC50 = 937 nM T64969 CZBA19 24905244 IC50 = 1200 nM T64969 CQ8OI1 24905246 IC50 = 45000 nM T64969 CIF2J5 24905251 IC50 = 3850 nM T64969 CPTE58 24905252 IC50 = 2120 nM T64969 CP50RD 24905280 IC50 = 1400 nM T64969 CG13ZM 24905281 IC50 = 33 nM T64969 CF0S6X 24905282 IC50 = 5950 nM T64969 C2Z5DN 24905285 IC50 = 12400 nM T64969 CL6GH8 24905286 IC50 = 100000 nM T64969 CKYO98 24905287 IC50 = 663 nM T64969 CRNQ65 24905288 IC50 = 2190 nM T64969 COD7I5 24905289 IC50 = 1670 nM T64969 C4LP7E 24905290 IC50 = 19000 nM T64969 CE9JC2 24905291 IC50 = 100000 nM T64969 C2GI1R 24905292 IC50 = 100000 nM T64969 CHW8C4 24905293 IC50 = 6450 nM T64969 CQF0H1 24905294 IC50 = 437 nM T64969 CNO7X0 24905295 IC50 = 158 nM T64969 C5WRG7 24905296 IC50 = 1400 nM T64969 CQ1S0U 24905297 IC50 = 5080 nM T64969 C4UES7 24905298 IC50 = 1160 nM T64969 CMS69P 24905299 IC50 = 2720 nM T64969 CC0U5M 24905300 IC50 = 67 nM T64969 CW7X6S 24905301 IC50 = 100000 nM T64969 C97IQV 24905302 IC50 = 318 nM T64969 CSJ47V 24905303 IC50 = 100000 nM T64969 CPN74C 24905304 IC50 = 9380 nM T64969 C5CS3N 24905305 IC50 = 2010 nM T64969 CK4XE9 24905307 IC50 = 100000 nM T64969 CTU6Z3 24905308 IC50 = 100000 nM T64969 C9SQX1 24905309 IC50 = 8700 nM T64969 CM75JP 24905310 IC50 = 15600 nM T64969 C9Q2BJ 24905311 IC50 = 12600 nM T64969 C9VUA1 24905312 IC50 = 12400 nM T64969 CU3RS1 24905313 IC50 = 17000 nM T64969 CYG3H2 24905314 IC50 = 2900 nM T64969 CV5Q7O 24905315 IC50 = 366 nM T64969 C8SA3O 24905316 IC50 = 270 nM T64969 CI5MN3 24905317 IC50 = 1580 nM T64969 CJ1P7K 24905318 IC50 = 1400 nM T64969 C1T6YQ 24905319 IC50 = 4800 nM T64969 CAU86X 24905320 IC50 = 2600 nM T64969 C54ISY 24905321 IC50 = 100000 nM T64969 C2GE5I 24905322 IC50 = 4800 nM T64969 C8D6YK 24905323 IC50 = 26000 nM T64969 C5NZH9 24905324 IC50 = 9140 nM T64969 C9D6JR 24905325 IC50 = 2900 nM T64969 CLZT41 24905326 IC50 = 1150 nM T64969 CW8FD3 24905327 IC50 = 775 nM T64969 CHB7A2 24905328 IC50 = 18000 nM T64969 CA8EI3 24905329 IC50 = 11000 nM T64969 CCQ0O7 24905330 IC50 = 6340 nM T64969 CJ81AS 24905331 IC50 = 100000 nM T64969 C8PW4H 24905332 IC50 = 324 nM T64969 C2Y5TF 24905333 IC50 = 236 nM T64969 CH9FL5 24905334 IC50 = 18000 nM T64969 C1S0PC 24905335 IC50 = 12000 nM T64969 C8N9MV 24905336 IC50 = 4320 nM T64969 C9E8BJ 24905338 IC50 = 100000 nM T64969 CX85AC 24905341 IC50 = 100000 nM T64969 CKZ80E 24905342 IC50 = 576 nM T64969 CO8SH1 24905343 IC50 = 3020 nM T64969 C7IZL6 24905344 IC50 = 100000 nM T64969 C5ZM4T 24936119 IC50 = 2400 nM T64969 C96GPD 24944848 IC50 = 7.1 nM T64969 CNMB03 24944849 IC50 = 7.8 nM T64969 CTCB27 24944850 IC50 = 9.4 nM T64969 C5PH0N 24944851 IC50 = 3.4 nM T64969 CK17HZ 24944855 IC50 = 8.2 nM T64969 C0BOJ2 24944856 IC50 = 7 nM T64969 CX05SV 24944930 IC50 = 3.1 nM T64969 CB8EZ0 24944934 IC50 = 15 nM T64969 C2CP6T 24944935 IC50 = 4.6 nM T64969 C1NZ8X 24945115 IC50 = 84.2 nM T64969 CF0U4T 24945204 IC50 = 10.4 nM T64969 C8W3YA 24945368 IC50 = 2.1 nM T64969 C2MYN7 24945689 IC50 = 9.08 nM T64969 C4V9GI 24960018 IC50 > 20000 nM T64969 C9B7PH 24970496 IC50 = 533 nM T64969 CGV1Q5 24970497 IC50 = 472 nM T64969 C4EG8R 24993189 IC50 > 10000 nM T64969 CHOK82 25000333 IC50 = 42 nM T64969 CBK82P 25011729 IC50 > 30000 nM T64969 CRO0Y8 25022735 IC50 = 122000 nM T64969 C72AJM 25022736 IC50 > 200000 nM T64969 CIK6V8 25025888 IC50 = 3.1 nM T64969 C0JGL8 25026082 IC50 = 3 nM T64969 CHY93R 25026085 IC50 = 8.8 nM T64969 C3DPS2 25026281 IC50 = 1.9 nM T64969 CD8IP2 25039251 IC50 = 12110 nM T64969 CHLQ49 25063262 IC50 = 30 nM T64969 C2KY1G 25094210 IC50 = 5048 nM T64969 C96EVA 25118036 IC50 = 8 nM T64969 CTV54O 25123227 IC50 > 10000 nM T64969 CG3XC9 25124150 IC50 = 57 nM T64969 CO2IR5 25124816 IC50 > 10000 nM T64969 C6BWZ8 25145145 IC50 > 100 nM T64969 C78YWA 25145716 IC50 > 500 nM T64969 CB21XV 25164469 Ki > 1800 nM T64969 CUX83H 25164675 Ki > 1800 nM T64969 C1H7BF 25164677 Ki > 1800 nM T64969 C6SD2A 25165081 Ki > 1800 nM T64969 C67TVH 25165085 Ki > 1800 nM T64969 CRJ6M7 25165279 Ki = 67 nM T64969 C7RBX0 25165280 Ki = 27 nM T64969 CPEY29 25165481 Ki = 17 nM T64969 C70DRX 25165482 Ki = 8 nM T64969 C6VZU2 25165861 Ki > 1800 nM T64969 CGUC69 25167072 Ki > 1800 nM T64969 CF4G1L 25167074 Ki > 1800 nM T64969 C35ZXL 25167075 Ki > 1800 nM T64969 C2D3FP 25167078 Ki > 1800 nM T64969 C37YSX 25167280 Ki > 1800 nM T64969 CX0O5A 25178331 IC50 = 9500 nM T64969 CIG4H0 25178539 IC50 = 4600 nM T64969 C4GI6J 25178540 IC50 = 9900 nM T64969 COB9G8 25181586 IC50 = 15070 nM T64969 CVY98J 25191769 Ki = 18 nM T64969 CP47JK 25192054 Ki = 43 nM T64969 C8K1YN 25192202 Ki = 290 nM T64969 C8TSW4 25192224 IC50 = 290 nM T64969 CBLF93 25192363 IC50 = 50 nM T64969 C09LAT 25192905 Ki = 49 nM T64969 CJ3YN8 25195273 IC50 = 12 nM T64969 C8NBA6 25195274 IC50 = 1 nM T64969 C6FGQ1 25206346 IC50 > 10000 nM T64969 C6XQB9 25207010 IC50 = 44 nM T64969 CRO09K 25211064 IC50 = 10 nM T64969 C8IJB9 25218207 IC50 = 10410 nM T64969 CR0FO4 25218688 EC50 = 335 nM T64969 CWNY70 25218689 EC50 = 742 nM T64969 CZ5M3A 25218690 EC50 = 520 nM T64969 CK9AO6 25218691 EC50 = 808 nM T64969 CXH7F8 25218692 EC50 = 85 nM T64969 CH2GL3 25218693 EC50 = 91 nM T64969 CU49HG 25218695 IC50 = 71 nM T64969 CU0YJ1 25218696 IC50 = 69 nM T64969 CQ6MZ0 25242463 IC50 = 54 nM T64969 CK7ZR2 25242643 IC50 = 320 nM T64969 CM31HJ 25263246 IC50 = 50 nM T64969 CAMY28 25263247 IC50 = 120 nM T64969 C6FB3N 25263248 IC50 = 2600 nM T64969 C7P4FS 25263249 IC50 = 1050 nM T64969 CV8Y5M 25263250 IC50 = 190 nM T64969 CKG21S 25263251 IC50 = 400 nM T64969 C7I4BG 25263252 IC50 = 280 nM T64969 C9TK3Q 25263253 IC50 = 180 nM T64969 CWE9C6 25263254 IC50 = 240 nM T64969 C9SL4P 25263255 IC50 = 1650 nM T64969 C4JQD8 25263256 IC50 = 630 nM T64969 CED02Z 25263257 IC50 = 80 nM T64969 CI79QB 25263258 IC50 = 30 nM T64969 C18VBO 25263259 IC50 = 33 nM T64969 CN89CY 25263260 IC50 = 120 nM T64969 C9JR3E 25263261 IC50 = 230 nM T64969 C0Y9TK 25263263 IC50 = 90 nM T64969 C5I4UQ 25263264 IC50 = 3160 nM T64969 CA0X9R 25263265 IC50 = 680 nM T64969 CW2J5P 25263266 IC50 = 240 nM T64969 CR7JS1 25263267 IC50 = 40 nM T64969 CT60US 25263268 IC50 = 50 nM T64969 C1NAD7 25263269 IC50 = 50 nM T64969 CJI43L 25263270 IC50 = 99 nM T64969 CANP37 25263271 IC50 = 63 nM T64969 CG3OH9 25263272 IC50 = 40 nM T64969 CZ0H9E 25263273 IC50 = 50 nM T64969 CY6HW8 25263274 IC50 = 40 nM T64969 C1WG7S 25263275 IC50 = 40 nM T64969 C6WV8D 25263276 IC50 = 125 nM T64969 CJW7I3 25263277 IC50 = 79 nM T64969 CTO10V 25263278 IC50 = 79 nM T64969 CZ4HN9 25263279 IC50 = 32 nM T64969 C7XEB3 25263280 IC50 = 79 nM T64969 C2ICK6 25263281 IC50 = 50 nM T64969 CZGQ83 25271178 IC50 = 41 nM T64969 CF2LZ7 25271179 IC50 = 150 nM T64969 CUAK50 25271517 IC50 = 76 nM T64969 CU09IM 26699441 IC50 = 50000 nM T64969 C69PNL 40433957 IC50 = 48600 nM T64969 CVM13K 42596931 IC50 = 42 nM T64969 CU53WB 42596953 IC50 = 18 nM T64969 CG2IJ8 42601891 IC50 < 1 nM T64969 C41TLH 42603880 IC50 = 35000 nM T64969 CS1AT2 42603881 IC50 = 93000 nM T64969 CZ2VH7 42604008 IC50 = 82000 nM T64969 CV1P3W 42604009 IC50 = 89000 nM T64969 CWS37O 42618140 IC50 > 10000 nM T64969 C2JV3O 42618143 IC50 > 10000 nM T64969 CG01BO 42618144 IC50 > 10000 nM T64969 CU9E4P 42629114 IC50 > 10000 nM T64969 CR5XJ4 42630202 IC50 = 7130 nM T64969 CJ5U1X 42639664 IC50 = 2.7 ug.mL-1 T64969 CPS5F6 43517028 IC50 = 6.2 nM T64969 CO42DC 44138048 IC50 > 10000 nM T64969 CL65QV 44138049 IC50 > 10000 nM T64969 CUX7D9 44143345 IC50 = 1000 nM T64969 C8YN5P 44143370 IC50 = 11000 nM T64969 C9CWO1 44143371 IC50 = 30000 nM T64969 C26XFL 44143372 IC50 = 22000 nM T64969 C5SEQ2 44143373 IC50 = 22000 nM T64969 CTN41Y 44156909 IC50 = 240 nM T64969 CN0X1C 44156917 IC50 = 63 nM T64969 CB0O2A 44186880 Ki > 1800 nM T64969 C9K7OP 44186882 Ki > 1800 nM T64969 CX0ZU8 44186885 Ki > 1800 nM T64969 CCFQ29 44187005 IC50 = 173 nM T64969 CNGV37 44189584 Ki > 1800 nM T64969 C2AV1K 44190762 IC50 = 2240 nM T64969 C6U2LF 44205208 IC50 = 4.1 nM T64969 CR03OF 44229775 IC50 = 2.9 nM T64969 CEL61X 44229839 IC50 = 2.6 nM T64969 C8DWO1 44229840 IC50 = 7 nM T64969 CNM3H2 44229841 IC50 = 21 nM T64969 C4NWP5 44246325 IC50 = 2200 nM T64969 C2EW0I 44246326 IC50 = 18200 nM T64969 CSD8T0 44246327 IC50 = 56500 nM T64969 CMKF08 44246328 IC50 = 13400 nM T64969 CAO87V 44246329 IC50 > 500000 nM T64969 CLU2V3 44246330 IC50 > 200000 nM T64969 CHZ6Q1 44269004 IC50 > 20000 nM T64969 C83QHW 44273476 IC50 > 100000 nM T64969 C8PT0I 44273491 IC50 > 200000 nM T64969 CS6NT3 44273526 IC50 = 100000 nM T64969 CG8H3R 44273527 IC50 > 200000 nM T64969 C7I1NX 44273528 IC50 = 95000 nM T64969 C3EFQ0 44273554 IC50 > 100000 nM T64969 CAJ48G 44273555 IC50 > 100000 nM T64969 C6VYU1 44273559 IC50 = 49000 nM T64969 C1WAE7 44273560 IC50 > 200000 nM T64969 CQEW06 44273561 IC50 > 200000 nM T64969 C82YSI 44273595 IC50 > 100000 nM T64969 CUG08T 44273597 IC50 > 200000 nM T64969 CIC13W 44273598 IC50 > 200000 nM T64969 CC8W2J 44273599 IC50 > 200000 nM T64969 CR1M9A 44273600 IC50 = 59000 nM T64969 CE6F2M 44273605 IC50 > 200000 nM T64969 CBV2Y3 44273617 IC50 > 200000 nM T64969 CAK08Y 44273618 IC50 = 90000 nM T64969 C0HG8U 44273619 IC50 = 75000 nM T64969 CMRX16 44273620 IC50 > 100000 nM T64969 CT79EW 44273623 IC50 > 200000 nM T64969 CZ6SM5 44273624 IC50 > 200000 nM T64969 CA8J9D 44273646 IC50 > 200000 nM T64969 C8JWQ2 44273647 IC50 = 180000 nM T64969 CI72SY 44273652 IC50 > 200000 nM T64969 CB0IL4 44273653 IC50 > 200000 nM T64969 CA6LH1 44273654 IC50 > 200000 nM T64969 C35TZW 44273659 IC50 > 100000 nM T64969 C8U2RI 44273699 IC50 > 200000 nM T64969 CY9LQ3 44273700 IC50 > 200000 nM T64969 CS7V9G 44278848 IC50 = 1.7 nM T64969 CIYC41 44279645 IC50 = 3762.4 nM T64969 CYEW69 44279647 IC50 = 2043.6 nM T64969 CMU95A 44285249 IC50 = 8.8 nM T64969 CO80RB 44285309 IC50 > 10000 nM T64969 CJQD03 44286273 IC50 = 350 nM T64969 CW02AS 44294903 IC50 > 50000 nM T64969 CRV54Q 44297168 IC50 = 11 nM T64969 C0RIG2 44297343 IC50 = 7 nM T64969 C5N7TD 44297358 IC50 = 120 nM T64969 C8ZAC4 44297408 IC50 = 4 nM T64969 CW0QU5 44299755 IC50 = 69 nM T64969 C2UZ3J 44299923 IC50 = 5 nM T64969 CT72NU 44299926 IC50 = 6 nM T64969 CD91OZ 44299938 IC50 = 5 nM T64969 CE2IC7 44299956 IC50 = 8 nM T64969 C72APV 44299983 IC50 = 8 nM T64969 C5ZSM3 44300005 IC50 = 2 nM T64969 C6CK9A 44300029 IC50 = 310 nM T64969 CFIO61 44300050 IC50 = 100 nM T64969 CJ7A3Y 44300081 IC50 = 8 nM T64969 CO25AL 44300251 IC50 = 35 nM T64969 CW6J2V 44313484 IC50 > 50000 nM T64969 C30GOH 44315116 IC50 = 17000 nM T64969 CA3C4I 44315117 IC50 > 50000 nM T64969 CMN04X 44315118 IC50 = 7000 nM T64969 CS8WZ6 44315309 IC50 = 40000 nM T64969 CUFQ79 44315416 IC50 = 55000 nM T64969 CKD14Y 44316725 IC50 = 1 nM T64969 CM2A1F 44316744 IC50 = 1 nM T64969 CLJ2P3 44316765 IC50 = 1 nM T64969 CK9L3S 44316797 IC50 = 7 nM T64969 C8IAY4 44316957 IC50 = 5 nM T64969 CD69PV 44317138 IC50 = 1 nM T64969 CY6P9K 44318047 IC50 = 70000 nM T64969 CSY8A3 44321301 IC50 = 19000 nM T64969 CCG2M5 44321317 IC50 = 9500 nM T64969 CY9ED1 44321395 IC50 > 100000 nM T64969 C5U1CR 44321686 IC50 > 10000 nM T64969 CETY53 44321717 IC50 > 100000 nM T64969 CV60ME 44321734 IC50 > 50000 nM T64969 C94MXP 44324651 IC50 = 170 nM T64969 CY48CU 44324654 IC50 = 430 nM T64969 C7T9RZ 44324666 IC50 = 730 nM T64969 CMP9D5 44324692 IC50 = 390 nM T64969 C9M3UO 44324693 IC50 = 11400 nM T64969 CB94OP 44324694 IC50 = 820 nM T64969 CI4P0C 44324869 IC50 = 300 nM T64969 CR5YP3 44324917 IC50 = 780 nM T64969 CSRW08 44324921 IC50 = 910 nM T64969 C7D6AQ 44324941 IC50 = 660 nM T64969 CL1QG5 44324942 IC50 = 10 nM T64969 CHKY38 44325074 IC50 = 27 nM T64969 CGHA16 44325116 IC50 = 65 nM T64969 CKC7R3 44330975 IC50 = 80500 nM T64969 CYT6F3 44330976 IC50 > 100000 nM T64969 CU58ZC 44331212 IC50 = 170 nM T64969 C2BSI9 44333736 IC50 = 3.3 nM T64969 C1KSW5 44335197 IC50 = 300 nM T64969 CB5J4A 44345182 IC50 = 4500 nM T64969 CW42OA 44345288 IC50 = 8709.64 nM T64969 C0A6IM 44345309 IC50 = 7943.28 nM T64969 CO9U4D 44345316 IC50 = 3400 nM T64969 C92MBY 44345327 IC50 = 3200 nM T64969 C5SMO1 44345334 IC50 = 48000 nM T64969 C57GUL 44345336 IC50 = 707.95 nM T64969 C09YJV 44345337 IC50 = 87000 nM T64969 CL73FP 44345342 IC50 = 15000 nM T64969 CCL45B 44345353 IC50 > 167000 nM T64969 CR5EL2 44345383 IC50 = 2000 nM T64969 CI02JL 44345396 IC50 = 4400 nM T64969 CHE2P1 44345431 IC50 = 900 nM T64969 CRQ76V 44345433 IC50 = 640 nM T64969 CJB1C4 44345439 IC50 = 5600 nM T64969 CVZ05R 44345469 IC50 = 6760.83 nM T64969 C0SH6O 44345633 IC50 = 14800 nM T64969 C06AQN 44345644 IC50 = 14454.4 nM T64969 CD62QG 44345647 IC50 = 5300 nM T64969 C2ESL8 44345648 IC50 = 12000 nM T64969 CW15XR 44345649 IC50 = 1700 nM T64969 CBC01N 44345675 IC50 > 50000 nM T64969 CPC35U 44345676 IC50 > 50000 nM T64969 C0KD4U 44346053 IC50 = 1100 nM T64969 CR1L3W 44346250 IC50 = 450000 nM T64969 C0D3UQ 44347328 IC50 = 9700 nM T64969 CJKU43 44347354 IC50 = 10300 nM T64969 C1QDI7 44347577 IC50 = 27200 nM T64969 C3WQ6J 44352770 IC50 = 910 nM T64969 C92FHZ 44352771 IC50 = 1300 nM T64969 CBX2L9 44352772 IC50 = 1100 nM T64969 CFJK28 44352785 IC50 = 7000 nM T64969 CF65DQ 44352791 IC50 > 100000 nM T64969 CL5QU9 44352816 IC50 = 3500 nM T64969 CKD32G 44352817 IC50 = 6400 nM T64969 CTZ3O4 44352818 IC50 = 1100 nM T64969 CRV1T2 44352826 IC50 = 160 nM T64969 CKGI05 44352842 IC50 = 110 nM T64969 C7YJ1S 44352843 IC50 = 7400 nM T64969 C8EVN3 44352844 IC50 = 3600 nM T64969 CI1R2S 44352845 IC50 > 70000 nM T64969 CQN85G 44352860 IC50 = 8180 nM T64969 CO43ND 44352873 IC50 = 13500 nM T64969 C2WRC4 44352890 IC50 = 4600 nM T64969 C1KO6C 44352905 IC50 = 12500 nM T64969 CK56AZ 44352914 IC50 = 4700 nM T64969 C2T4XV 44352915 IC50 = 8180 nM T64969 CX1SD9 44352928 IC50 = 2400 nM T64969 CIUR28 44352929 IC50 = 1300 nM T64969 CJE57B 44352930 IC50 = 4800 nM T64969 C84FIH 44352951 IC50 = 2600 nM T64969 CVHA74 44352970 IC50 = 260 nM T64969 CQ2F5D 44352972 IC50 = 17 nM T64969 CX82RD 44352973 IC50 = 220 nM T64969 COZ52V 44353100 IC50 = 31 nM T64969 CLX76Q 44353115 IC50 = 19 nM T64969 C9RUC6 44353122 IC50 = 330 nM T64969 CUG68J 44353130 IC50 = 43 nM T64969 C50EHA 44353341 IC50 > 100000 nM T64969 CP8B0J 44353452 IC50 > 100000 nM T64969 CQZM34 44355143 IC50 > 20000 nM T64969 CX1I0D 44355168 IC50 > 1000 nM T64969 C2F9DZ 44355323 IC50 > 20000 nM T64969 C4LKS3 44355443 IC50 = 100 nM T64969 CJWK61 44355456 IC50 > 50000 nM T64969 C9YI1R 44355486 IC50 = 10 nM T64969 CM0BW2 44355543 IC50 > 50000 nM T64969 C0VSJ3 44355545 IC50 > 20000 nM T64969 CIV6A3 44355618 IC50 = 12000 nM T64969 CYR4C8 44355673 IC50 > 50000 nM T64969 CM24OQ 44355891 IC50 > 20000 nM T64969 CHL4V6 44355892 IC50 > 20000 nM T64969 CM6X3O 44355907 IC50 = 1300 nM T64969 C30OUK 44355908 IC50 = 7000 nM T64969 CX0R3O 44355931 IC50 > 50000 nM T64969 CK4U5B 44361553 IC50 = 1698.24 nM T64969 CM56JY 44361640 IC50 = 3019.95 nM T64969 CT2R7Z 44361668 IC50 = 15848.93 nM T64969 C5RZI9 44361703 IC50 = 19054.61 nM T64969 C04PXM 44361706 IC50 = 47863.01 nM T64969 C1NRF6 44361710 IC50 = 53703.18 nM T64969 CAZD14 44361915 IC50 = 165958.69 nM T64969 CFY75E 44363476 IC50 = 2100 nM T64969 C1FM7A 44367247 IC50 = 2.7 nM T64969 CSW63A 44367400 IC50 > 10000 nM T64969 CWJ61S 44367436 IC50 = 33 nM T64969 C0RBE5 44367446 IC50 = 85 nM T64969 CQL29S 44367457 IC50 = 9.4 nM T64969 C9GX4S 44367566 IC50 = 40 nM T64969 CYV2D7 44368815 IC50 > 10000 nM T64969 C10VDK 44371971 IC50 = 330 nM T64969 C2GRI5 44372004 IC50 = 10 nM T64969 C9NYG0 44372005 IC50 = 110 nM T64969 CFM6C8 44372022 IC50 = 8 nM T64969 CCGX21 44372180 IC50 = 35 nM T64969 C6L4CX 44372197 IC50 = 82 nM T64969 CSA68M 44372283 IC50 = 540 nM T64969 C8RL0S 44377259 IC50 = 3.9 nM T64969 CC3T6E 44381073 IC50 = 13200 nM T64969 CQT59Y 44381095 IC50 = 9700 nM T64969 C8LZ0Q 44381185 IC50 = 600 nM T64969 C6FCU8 44381190 IC50 = 440 nM T64969 C1D2LU 44381191 IC50 = 830 nM T64969 CJZD30 44381192 IC50 = 740 nM T64969 CFQ57C 44381224 IC50 = 570 nM T64969 CZ64TC 44381237 IC50 = 80 nM T64969 C5WQY2 44381238 IC50 = 250 nM T64969 CD0WU4 44381266 IC50 = 420 nM T64969 C7VJ9M 44381267 IC50 = 2820 nM T64969 C9S1EJ 44381268 IC50 = 790 nM T64969 CM64RL 44381269 IC50 = 300 nM T64969 CBKP57 44381381 IC50 = 450 nM T64969 C2DCJ0 44381398 IC50 = 8300 nM T64969 C6LSB4 44381409 IC50 = 295 nM T64969 CE7H4L 44381435 IC50 = 500 nM T64969 C98OGL 44381436 IC50 = 330 nM T64969 CEQ7M0 44381445 IC50 = 930 nM T64969 CWKB67 44381507 IC50 = 14400 nM T64969 CX98KS 44381508 IC50 = 440 nM T64969 C6LC8M 44381556 IC50 = 310 nM T64969 CCA56B 44381571 IC50 = 1470 nM T64969 C5Z9MJ 44381580 IC50 = 750 nM T64969 CY58LS 44381608 IC50 = 2100 nM T64969 C6DQX7 44381674 IC50 = 2200 nM T64969 C75NGL 44384514 IC50 = 1300 nM T64969 CV0F4D 44384547 IC50 = 12000 nM T64969 CQF8Y7 44384548 IC50 = 1100 nM T64969 CF01AV 44384717 IC50 = 5300 nM T64969 CI2L9R 44384964 IC50 = 6400 nM T64969 CC09FT 44384965 IC50 = 1400 nM T64969 CE9PU7 44385035 IC50 = 6400 nM T64969 CQGW07 44385080 IC50 = 700 nM T64969 CL4Y9M 44385116 IC50 = 800 nM T64969 CUI34C 44385739 IC50 = 2650 nM T64969 C87MAJ 44388483 IC50 = 72 nM T64969 CB7QM3 44388486 IC50 = 151 nM T64969 C6WDG3 44388487 IC50 = 210 nM T64969 C3YM9F 44388494 IC50 = 255 nM T64969 CN4L2V 44388499 IC50 = 247 nM T64969 CUA90G 44388501 IC50 = 400 nM T64969 CBU34A 44389468 IC50 = 26 nM T64969 CU9Z5Y 44395043 IC50 = 490 nM T64969 CF31XZ 44395044 IC50 > 33000 nM T64969 CCLX29 44395123 IC50 = 2800 nM T64969 CCAI71 44395145 IC50 > 33000 nM T64969 CZ97PV 44395162 IC50 = 2200 nM T64969 CZ6HP1 44395171 IC50 = 11000 nM T64969 C2T6DH 44395178 IC50 = 29000 nM T64969 C0XQ2Z 44395209 IC50 > 33000 nM T64969 CTDI68 44395241 IC50 > 33000 nM T64969 CW3BP8 44398371 IC50 = 45800 nM T64969 CH9NR8 44403081 IC50 = 200 nM T64969 C0AR9C 44403420 IC50 = 5 nM T64969 CGQ26K 44403425 IC50 = 1800 nM T64969 CRV6B4 44403429 IC50 = 2400 nM T64969 CTY5K7 44403435 IC50 = 2100 nM T64969 C47XFZ 44403436 IC50 = 440 nM T64969 C8K4AL 44407237 IC50 = 12600 nM T64969 CUA18B 44407238 IC50 = 31000 nM T64969 C04HFE 44407248 IC50 > 50000 nM T64969 CR3O1C 44407275 IC50 = 5100 nM T64969 C70BFV 44407276 IC50 = 13600 nM T64969 CMH7W6 44407277 IC50 = 9000 nM T64969 CIQR47 44409038 IC50 = 1700 nM T64969 C6UE2S 44409043 IC50 = 3700 nM T64969 C64ZYA 44409055 IC50 = 3400 nM T64969 CY1AQ7 44409056 IC50 = 7000 nM T64969 CT9M4U 44409118 IC50 = 873 nM T64969 C46NPW 44409144 IC50 = 225 nM T64969 C6E4QU 44409147 IC50 = 1000 nM T64969 C29RFN 44409148 IC50 = 9601 nM T64969 C9H3VZ 44409149 IC50 = 671 nM T64969 C4V6FS 44409152 IC50 > 10000 nM T64969 CW24DU 44409153 IC50 = 5400 nM T64969 C4S6ZN 44409156 IC50 = 4900 nM T64969 C3HFY0 44409208 IC50 = 3 nM T64969 CW87XM 44409211 IC50 = 66 nM T64969 CHD92U 44409225 IC50 = 2000 nM T64969 CNS1X6 44409226 IC50 = 9800 nM T64969 CIX8D6 44409229 IC50 > 10000 nM T64969 C2MN0X 44409230 IC50 > 10000 nM T64969 CNQL75 44409263 IC50 = 1000 nM T64969 C7G6OS 44409281 IC50 > 10000 nM T64969 C0TNV5 44409288 IC50 < 2 nM T64969 C8UN1W 44409346 IC50 = 1000 nM T64969 CQW9E1 44409347 IC50 = 10 nM T64969 C03UCB 44409353 IC50 = 4400 nM T64969 C7W8VG 44409387 IC50 = 1384 nM T64969 C9SP0E 44409388 IC50 < 2 nM T64969 CM1D9O 44409422 IC50 = 187 nM T64969 CZQ03C 44409423 IC50 = 8068 nM T64969 C7HD4Q 44410411 IC50 = 320 nM T64969 CED5S6 44410414 IC50 = 85 nM T64969 C0A7XB 44410560 IC50 = 63 nM T64969 C5WKG0 44410574 IC50 = 25100 nM T64969 CDQ4S6 44410648 IC50 = 42 nM T64969 C4OJ1S 44410700 IC50 = 110 nM T64969 CIY53K 44410704 IC50 = 79 nM T64969 CPH17L 44410710 IC50 = 50 nM T64969 C2J1KU 44410716 IC50 = 31 nM T64969 CV09DY 44410717 IC50 = 8 nM T64969 CP3CI1 44410720 IC50 = 50 nM T64969 C8W7AD 44410723 IC50 = 40 nM T64969 CAT5X4 44410829 IC50 = 300 nM T64969 CC6Y5P 44410844 IC50 = 300 nM T64969 CG34TY 44410851 IC50 = 70 nM T64969 C41EIA 44410869 IC50 = 10 nM T64969 CB6AE8 44410948 IC50 = 70 nM T64969 CXZG12 44410949 IC50 < 1 nM T64969 CS7IE9 44410953 IC50 = 100 nM T64969 CA9M4X 44410954 IC50 = 90 nM T64969 C3SP5H 44410955 IC50 = 450 nM T64969 C5D6YP 44410956 IC50 = 10 nM T64969 C5W1VC 44410959 IC50 = 130 nM T64969 CM1C2G 44410960 IC50 = 30 nM T64969 CVSI80 44411048 IC50 = 80 nM T64969 CN72BR 44411161 IC50 = 50 nM T64969 C4AW0O 44411183 IC50 = 25 nM T64969 C0XJC3 44412177 IC50 = 1693 nM T64969 C5QD2S 44412181 IC50 = 81 nM T64969 CRH3Y6 44412244 IC50 = 156 nM T64969 C7KZV2 44414322 IC50 > 50000 nM T64969 CJM06T 44414347 IC50 > 50000 nM T64969 C16IVC 44416188 IC50 = 50 nM T64969 COFI73 44416243 IC50 = 16 nM T64969 CS8U4Y 44416288 IC50 = 19 nM T64969 CVA3S4 44416289 IC50 = 17 nM T64969 CD4H3O 44416334 IC50 = 62900 nM T64969 CO25JT 44416335 IC50 = 14100 nM T64969 C1KW2L 44416347 IC50 > 100000 nM T64969 CMG28W 44416407 IC50 = 51 nM T64969 C5R7IW 44416429 IC50 = 7400 nM T64969 C7C4TK 44416433 IC50 = 6100 nM T64969 C0IUL9 44416434 IC50 = 4600 nM T64969 CUBA46 44416461 IC50 = 18 nM T64969 CR42NY 44416467 IC50 = 10800 nM T64969 C5XE7I 44416473 IC50 = 15200 nM T64969 CAP9S0 44416499 IC50 = 24600 nM T64969 C41SAP 44416508 IC50 = 3400 nM T64969 CA83EK 44416509 IC50 = 8200 nM T64969 CK8R2O 44416545 IC50 = 1200 nM T64969 CX17JM 44416560 IC50 = 150 nM T64969 CD2FC0 44416568 IC50 = 5600 nM T64969 CPIA51 44416569 IC50 > 100000 nM T64969 C7QH2K 44416595 IC50 = 114 nM T64969 CX3DU9 44416596 IC50 > 100000 nM T64969 CYU1W9 44416603 IC50 = 17000 nM T64969 C7DTI2 44416610 IC50 < 0.5 nM T64969 CJS8C5 44416611 IC50 = 9 nM T64969 C0CQ4S 44416612 IC50 = 1 nM T64969 C35BCH 44416635 IC50 = 300 nM T64969 CO9MX1 44416647 IC50 = 14500 nM T64969 C6HQ5D 44416655 IC50 = 1100 nM T64969 CIY3J4 44416673 IC50 = 9 nM T64969 CIV18H 44416687 IC50 = 300 nM T64969 C43VZI 44416688 IC50 = 800 nM T64969 CF5UH3 44416692 IC50 = 900 nM T64969 C43NYR 44416693 IC50 = 8700 nM T64969 C8RHO3 44416712 IC50 = 200 nM T64969 C2L0ZB 44416719 IC50 = 106 nM T64969 CZ3WQ2 44416741 IC50 = 7100 nM T64969 CAV3B1 44417449 IC50 > 3000 nM T64969 CKD97C 44417487 IC50 > 3000 nM T64969 COPG94 44427519 IC50 > 10000 nM T64969 C0PLD7 44428887 IC50 = 283.3 nM T64969 C2V1FP 44428888 IC50 = 43.1 nM T64969 C2UT9G 44428889 IC50 = 166.7 nM T64969 C8XRO1 44428890 IC50 = 18.7 nM T64969 C3A2HC 44428891 IC50 = 791.9 nM T64969 C42KHG 44428893 IC50 = 35.6 nM T64969 CDE73U 44428895 IC50 = 295.2 nM T64969 C5H3DV 44428898 IC50 = 107.3 nM T64969 C2V1ER 44428899 IC50 = 173.1 nM T64969 CLGZ52 44428901 IC50 < 10 nM T64969 C8LI7S 44428906 IC50 = 7710 nM T64969 C7BZ0K 44430019 IC50 = 81 nM T64969 CJ1U9R 44430027 IC50 = 1000 nM T64969 COBA27 44430030 IC50 = 140 nM T64969 C8WJV9 44430032 IC50 = 130 nM T64969 C9UYP5 44430034 IC50 = 26 nM T64969 CQ67VA 44430037 IC50 = 190 nM T64969 CW58IO 44430039 IC50 = 130 nM T64969 CA98KR 44432441 IC50 > 6000 nM T64969 C5QJ0K 44435405 IC50 < 5000 nM T64969 CNSW23 44435406 IC50 > 40000 nM T64969 CIOY17 44435407 IC50 > 40000 nM T64969 CCV5A0 44435408 IC50 > 40000 nM T64969 C73EMA 44435409 IC50 > 40000 nM T64969 CAJ5W6 44435435 IC50 > 40000 nM T64969 CX09ZA 44440812 IC50 = 210 nM T64969 C36FXV 44440815 IC50 = 86 nM T64969 CF5UR8 44440816 IC50 = 200 nM T64969 C87FRB 44440817 IC50 = 1800 nM T64969 CNCU91 44440820 IC50 = 340 nM T64969 CL1N3P 44440821 IC50 = 490 nM T64969 C85SOF 44440823 IC50 = 30 nM T64969 C8GHB0 44440824 IC50 = 460 nM T64969 C74ONA 44440826 IC50 = 140 nM T64969 CNU0P1 44440830 IC50 = 130 nM T64969 CU72VL 44440831 IC50 = 190 nM T64969 CNY07A 44440833 IC50 = 83 nM T64969 CZ4G2C 44440835 IC50 = 640 nM T64969 C85HCV 44440836 IC50 = 210 nM T64969 CO6DP3 44440837 IC50 = 560 nM T64969 C4Y1TD 44440839 IC50 = 500 nM T64969 CWC9V6 44440840 IC50 = 810 nM T64969 CIF14K 44440841 IC50 = 120 nM T64969 CJ23DP 44440842 IC50 = 690 nM T64969 CO8WZ7 44440843 IC50 = 68 nM T64969 CJL0G8 44440844 IC50 = 400 nM T64969 CA75PM 44440874 IC50 = 430 nM T64969 CAM78I 44441000 IC50 = 50 nM T64969 C6ZEJ5 44441012 IC50 = 190 nM T64969 C3MW6G 44441013 IC50 = 40 nM T64969 C3AZF8 44441014 IC50 = 47 nM T64969 CJC06N 44441015 IC50 = 190 nM T64969 CWJ1U3 44441016 IC50 = 530 nM T64969 C2IL0Y 44441017 IC50 = 19 nM T64969 CMW7T5 44442025 IC50 = 3 nM T64969 C3U1GC 44442026 IC50 = 2580 nM T64969 C9J2FM 44442027 IC50 = 2 nM T64969 CU7N0D 44442028 IC50 = 191 nM T64969 C8OSC2 44442129 IC50 = 331 nM T64969 CN0PD8 44442133 IC50 = 1640.6 nM T64969 CH4T0Y 44442137 IC50 = 185.8 nM T64969 CX2F5J 44442142 IC50 = 114.2 nM T64969 C4LNA9 44442145 IC50 = 94.5 nM T64969 CLD6A1 44442146 IC50 = 151.5 nM T64969 CKBP38 44442147 IC50 = 50.3 nM T64969 CDT1F0 44442149 IC50 = 88.7 nM T64969 C5ETZ9 44442150 IC50 = 921 nM T64969 CZKI61 44442152 IC50 = 402.1 nM T64969 CC06RB 44442154 IC50 = 1362.6 nM T64969 CGY4Q2 44442155 IC50 = 205.8 nM T64969 C8CIJ2 44442169 IC50 = 13 nM T64969 C36JSL 44442170 IC50 = 80 nM T64969 CD3LW7 44442179 IC50 = 4 nM T64969 C8LY2G 44442184 IC50 = 10 nM T64969 CPQ02C 44442185 IC50 = 12 nM T64969 CGFL71 44442186 IC50 = 1.8 nM T64969 CEX85R 44442187 IC50 = 11.7 nM T64969 CY61BH 44442188 IC50 = 4.2 nM T64969 C5JRD8 44442189 IC50 = 662 nM T64969 C5R4QE 44442729 Ki = 24 nM T64969 CGC76I 44442730 Ki = 180 nM T64969 CJM6N5 44442731 Ki = 360 nM T64969 CH2FS6 44442732 Ki = 120 nM T64969 CZ7FC6 44442733 Ki = 64 nM T64969 C6PNZ4 44442734 Ki = 52 nM T64969 C8N1EQ 44442735 Ki = 68 nM T64969 C26EVP 44442736 IC50 = 173 nM T64969 C0S6PN 44442737 IC50 = 52.8 nM T64969 CAZ5O7 44442738 IC50 = 5 nM T64969 CM9XW1 44442739 Ki = 360 nM T64969 CFOH51 44442740 Ki = 340 nM T64969 CX10DZ 44442742 Ki = 40 nM T64969 CN12IA 44442744 Ki = 400 nM T64969 C0DOP6 44442745 Ki = 80 nM T64969 CJ4BV0 44442747 Ki = 44 nM T64969 CJHV89 44442752 Ki = 80 nM T64969 CYS18W 44442753 Ki = 220 nM T64969 C26GVA 44442758 Ki = 52 nM T64969 CZG61W 44442759 Ki = 36 nM T64969 C4YMI9 44447890 IC50 > 1000 nM T64969 CR65PM 44447895 IC50 > 1000 nM T64969 CR62KV 44448938 IC50 = 267 nM T64969 CT9R7H 44448969 IC50 = 306 nM T64969 C9RV4Q 44448995 IC50 = 1123 nM T64969 CUB12D 44449577 IC50 = 150 nM T64969 CSA12W 44450544 IC50 = 5000000 nM T64969 C3ZBV8 44450546 IC50 = 13300 nM T64969 C0C2RS 44450792 IC50 = 780 nM T64969 C0MXV2 44450803 IC50 > 10000 nM T64969 C7HIM2 44452543 IC50 > 500 nM T64969 CZ9H4D 44452544 IC50 > 500 nM T64969 CQ1M7K 44455194 IC50 < 1 nM T64969 C86DQE 44455195 IC50 = 28 nM T64969 C20ISD 44455293 IC50 = 13 nM T64969 CUN90T 44455330 IC50 = 18 nM T64969 CNR2V1 44456900 IC50 = 3.236 nM T64969 C3AWN6 44456909 IC50 = 1.514 nM T64969 CBD75X 44456910 IC50 = 40.74 nM T64969 CAM6P8 44456911 IC50 = 4786.3 nM T64969 CVYZ16 44456912 IC50 = 3715.35 nM T64969 C7GQR6 44456927 IC50 = 0.912 nM T64969 C6S5YU 44456928 IC50 = 8.511 nM T64969 CHE0Q7 44456929 IC50 = 25.7 nM T64969 C7J4MG 44456940 IC50 = 0.5129 nM T64969 CD18RN 44456941 IC50 = 245.47 nM T64969 CIWS70 44456942 IC50 = 10 nM T64969 C1MI8R 44456962 IC50 = 7.413 nM T64969 C3P2SB 44456963 IC50 = 40.74 nM T64969 CAF3L1 44456987 IC50 = 7.244 nM T64969 CLW80I 44456989 IC50 = 251.19 nM T64969 CF1UQ0 44457004 IC50 = 45.71 nM T64969 C93BJI 44457005 IC50 = 8.913 nM T64969 CJB04A 44457006 IC50 = 39.81 nM T64969 C7B2RU 44457007 IC50 = 13.18 nM T64969 CAF6E5 44457023 IC50 = 12.02 nM T64969 C7FE2H 44457024 IC50 = 1.202 nM T64969 CVB57O 44457026 IC50 = 3.236 nM T64969 C8K3BG 44457027 IC50 = 14.13 nM T64969 C5MFW9 44457038 IC50 = 0.9333 nM T64969 C0R5SP 44457039 IC50 = 0.2455 nM T64969 C9XD8N 44457040 IC50 = 2.63 nM T64969 C8I0UN 44457041 IC50 = 29.51 nM T64969 CDK0Q7 44457055 IC50 = 9.333 nM T64969 C0P7JH 44457062 IC50 = 3.548 nM T64969 CQF2J4 44457064 IC50 = 9.333 nM T64969 C3JX0B 44457065 IC50 = 5.623 nM T64969 C8ZG4J 44457066 IC50 = 5.495 nM T64969 CB7Z4F 44457080 IC50 = 1.413 nM T64969 C2R4QL 44457083 IC50 = 16.22 nM T64969 C5G2UO 44457084 IC50 = 0.2818 nM T64969 C24HUL 44457085 IC50 = 2.344 nM T64969 C63CIA 44457086 IC50 = 5.012 nM T64969 CI39XF 44457115 IC50 = 5.495 nM T64969 CR06HM 44457116 IC50 = 40.74 nM T64969 CDV1E5 44457117 IC50 = 120.23 nM T64969 C5Y7HJ 44457118 IC50 = 70.79 nM T64969 C1PWV8 44457132 IC50 = 0.6166 nM T64969 C62QBG 44457133 IC50 = 1.905 nM T64969 C49BNA 44457135 IC50 = 4897.79 nM T64969 C35NVA 44457136 IC50 = 851.14 nM T64969 C9FMH7 44457137 IC50 = 1819.7 nM T64969 CU1I4O 44457148 IC50 = 676.08 nM T64969 CZ1R3H 44457149 IC50 = 131.83 nM T64969 CL0P5W 44471009 IC50 = 0.22 nM T64969 CAS03E 44481081 IC50 = 1340 nM T64969 C4TF5E 44481332 IC50 = 1760 nM T64969 C9D2SF 44515230 IC50 = 270 nM T64969 C5RA7I 44515232 IC50 = 850 nM T64969 CYH6P3 44520205 IC50 = 2090 nM T64969 CDFI53 44528870 IC50 = 68 nM T64969 CI8X2C 44528924 IC50 = 4 nM T64969 C9ZU2D 44528930 IC50 = 138 nM T64969 CXR98Y 44528960 IC50 = 6 nM T64969 CI3JR0 44532526 IC50 > 50000 nM T64969 CFP97X 44532811 IC50 = 3 nM T64969 C0LY6E 44552561 EC50 > 10000 nM T64969 C7KRU3 44552562 IC50 > 10000 nM T64969 CRPM76 44555376 IC50 = 200 nM T64969 C3JUM4 44555383 IC50 = 630 nM T64969 CYV71I 44555430 IC50 = 15.5 nM T64969 C3VRO9 44557921 IC50 > 10000 nM T64969 C1A4XG 44562420 IC50 = 458 nM T64969 C3UV2W 44562431 IC50 = 620 nM T64969 C5AS8P 44564023 IC50 = 1.514 nM T64969 CA8E5X 44564024 IC50 = 19.95 nM T64969 C68VDI 44564025 IC50 = 6.607 nM T64969 CPO8W9 44564026 IC50 = 0.912 nM T64969 C1K6BV 44564031 IC50 = 0.1698 nM T64969 CYE06Q 44564061 IC50 = 1.585 nM T64969 C93BFU 44564062 IC50 = 1.202 nM T64969 CLAF15 44564063 IC50 = 0.5012 nM T64969 C2T8PE 44564064 IC50 = 0.5495 nM T64969 CX2Q1J 44564065 IC50 = 0.6918 nM T64969 CX4M3C 44564100 IC50 = 1.738 nM T64969 COSJ65 44564101 IC50 = 1.096 nM T64969 CLYD65 44564102 IC50 = 1.585 nM T64969 C9BA2G 44564103 IC50 = 9.12 nM T64969 CD5QH9 44564104 IC50 = 1.202 nM T64969 C8G6MO 44564165 IC50 = 0.7079 nM T64969 CIW9B5 44564166 IC50 = 44.67 nM T64969 CN4WY6 44564167 IC50 = 26.92 nM T64969 CN0AS3 44564168 IC50 = 0.3715 nM T64969 C59GKR 44564169 IC50 = 2.692 nM T64969 CW13TY 44564170 IC50 = 1.514 nM T64969 CC17KX 44564171 IC50 = 4.169 nM T64969 CX0US9 44564172 IC50 = 2.692 nM T64969 C0TUR8 44564191 IC50 = 3.311 nM T64969 CD45HS 44564192 IC50 = 2.399 nM T64969 C4VQP9 44564193 IC50 = 0.4365 nM T64969 C81WPX 44564194 IC50 = 1.096 nM T64969 COQ61X 44564233 IC50 = 0.7244 nM T64969 C0Y2WH 44564234 IC50 = 0.8128 nM T64969 CPLB92 44564235 IC50 = 0.5623 nM T64969 C1KWB4 44564236 IC50 = 1.445 nM T64969 C04JAC 44564270 IC50 = 93.33 nM T64969 C9VAI7 44564303 IC50 = 0.4467 nM T64969 CXI08J 44564304 IC50 = 0.537 nM T64969 C2DS5N 44564306 IC50 = 8.6 nM T64969 CM3J7B 44564307 IC50 = 6 nM T64969 CP9RO4 44564308 IC50 = 8 nM T64969 CF41OU 44564309 IC50 = 8 nM T64969 CQ0ID4 44564335 IC50 < 1 nM T64969 CAE13O 44564361 IC50 = 1.096 nM T64969 C59TUM 44564362 IC50 = 1.202 nM T64969 C4ZTX0 44564365 IC50 = 10320 nM T64969 C1QFI4 44564394 IC50 = 1.698 nM T64969 CZCF57 44564395 IC50 = 3.631 nM T64969 CXFP58 44564396 IC50 = 3.89 nM T64969 C5VO9D 44564397 IC50 = 3.02 nM T64969 C29OUL 44564398 IC50 = 3.715 nM T64969 CFU1Q8 44564399 IC50 = 0.4365 nM T64969 CD10EC 44564400 IC50 = 5390 nM T64969 CF1T5K 44564401 IC50 = 13570 nM T64969 CD6XJ4 44564402 IC50 = 5220 nM T64969 C7OU0D 44564403 IC50 = 10590 nM T64969 CYD0K8 44564435 IC50 = 0.7762 nM T64969 CS92EV 44564436 IC50 = 0.4169 nM T64969 C41PEW 44564437 IC50 = 1.995 nM T64969 C4CH2U 44564438 IC50 = 1.514 nM T64969 C58LAW 44564439 IC50 = 0.6918 nM T64969 C27UGT 44564440 IC50 = 0.7943 nM T64969 CNQE26 44564441 IC50 = 1.585 nM T64969 C8UR0S 44564442 IC50 = 40.74 nM T64969 CZ1LX2 44564443 IC50 = 20.89 nM T64969 C2PTY9 44564444 IC50 = 3.715 nM T64969 C6NB0I 44564445 IC50 = 7500 nM T64969 CLR6X7 44564476 IC50 = 1.82 nM T64969 CEUJ39 44564477 IC50 = 0.7586 nM T64969 COR0K6 44564478 IC50 = 1.514 nM T64969 C5P0CL 44564479 IC50 = 1.698 nM T64969 CV67XP 44564480 IC50 = 8.71 nM T64969 CO6C8D 44564481 IC50 = 5.129 nM T64969 C91WOF 44564482 IC50 = 4.786 nM T64969 CB1O0P 44564526 IC50 = 0.7586 nM T64969 C4T3PW 44564527 IC50 = 0.1585 nM T64969 CR2J8L 44564528 IC50 = 2.692 nM T64969 C3NMY1 44564529 IC50 = 0.955 nM T64969 CXD0W8 44564530 IC50 = 0.9772 nM T64969 CC62JT 44564704 IC50 = 150 nM T64969 CC7E4K 44564705 IC50 > 10000 nM T64969 C42ZEW 44564706 IC50 = 2000 nM T64969 C53MCK 44564747 IC50 > 10000 nM T64969 CDI31F 44564748 IC50 > 10000 nM T64969 CA17NT 44564749 IC50 > 10000 nM T64969 CMIZ20 44564750 IC50 > 10000 nM T64969 CSO9F8 44564751 IC50 > 10000 nM T64969 C8ATG9 44564787 IC50 > 10000 nM T64969 CM50GS 44564788 IC50 > 10000 nM T64969 C3Q0DX 44564789 IC50 = 1300 nM T64969 CP40XB 44564790 IC50 = 720 nM T64969 C35NTB 44564791 IC50 = 7700 nM T64969 CJY83G 44564817 IC50 = 5100 nM T64969 CLK98G 44564818 IC50 = 7800 nM T64969 CF2D1K 44564819 IC50 = 2600 nM T64969 C3CQ9K 44564820 IC50 > 10000 nM T64969 CI8V2L 44564821 IC50 > 10000 nM T64969 C9PO7J 44564860 IC50 > 10000 nM T64969 C16FJW 44564861 IC50 > 10000 nM T64969 C8AMX5 44564862 IC50 = 5300 nM T64969 CTR59U 44564863 IC50 > 10000 nM T64969 C9EY4C 44564864 IC50 = 800 nM T64969 CG5Z7T 44564910 IC50 > 10000 nM T64969 CU9O4C 44564911 IC50 > 10000 nM T64969 CXZ15S 44564954 IC50 > 10000 nM T64969 CZ78WJ 44564955 IC50 > 10000 nM T64969 CJ1X9V 44565013 IC50 = 1900 nM T64969 CN2Q3D 44565014 IC50 = 3300 nM T64969 CM2GN3 44565015 IC50 > 10000 nM T64969 C6RV9I 44565016 IC50 = 1700 nM T64969 CJC85A 44565069 IC50 = 1600 nM T64969 CSOH56 44565943 IC50 > 200000 nM T64969 CTUD59 44565958 IC50 > 200000 nM T64969 C6IFZ9 44565965 IC50 > 200000 nM T64969 CRX0M5 44571414 IC50 = 304 nM T64969 C9KY2N 44571415 IC50 = 115 nM T64969 CT92ZI 44571431 IC50 = 10 nM T64969 C0W9NE 44571432 IC50 = 4 nM T64969 CKY57M 44571433 IC50 = 8 nM T64969 C2RQ3H 44571434 IC50 = 7 nM T64969 CUCI91 44571435 IC50 = 15 nM T64969 C7LVG6 44571436 IC50 = 54 nM T64969 CIU14N 44571437 IC50 = 121 nM T64969 CLP71D 44571448 IC50 = 2 nM T64969 CEIK76 44571449 IC50 = 5 nM T64969 CFNT92 44571450 IC50 = 3 nM T64969 CIB7R5 44571451 IC50 = 3 nM T64969 CK6L2W 44571452 IC50 = 68 nM T64969 CI1PL5 44571453 IC50 = 9 nM T64969 CZ0ID1 44571454 IC50 = 96 nM T64969 CWFB42 44571820 IC50 = 22 nM T64969 CU9Y0V 44576127 IC50 = 0.9 ug.mL-1 T64969 CPKL09 44576144 IC50 = 800 nM T64969 CG4E2Z 44576145 IC50 = 600 nM T64969 CI87PR 44576146 IC50 = 3000 nM T64969 C2U7IW 44576150 IC50 = 6000 nM T64969 C8ST7I 44576151 IC50 = 900000 nM T64969 C3K5AT 44576152 IC50 = 10000 nM T64969 CI8J1E 44576153 IC50 = 10000 nM T64969 CD0AC6 44576154 IC50 = 400000 nM T64969 C35DJE 44576155 IC50 = 600000 nM T64969 C9YXF6 44576156 IC50 = 600000 nM T64969 C4KBE3 44576157 IC50 = 1000 nM T64969 CQL4X2 44576163 IC50 = 10000 nM T64969 C7Q1VU 44580077 IC50 > 25000 nM T64969 CL90SE 44580358 IC50 > 25000 nM T64969 CK1VE7 44580420 IC50 > 25000 nM T64969 CH2R7X 44580449 IC50 > 25000 nM T64969 C1VH0C 44580532 IC50 > 25000 nM T64969 CXC52J 44580649 IC50 > 25000 nM T64969 CE32BQ 44580689 IC50 = 700 nM T64969 C8Z5AX 44580778 IC50 > 25000 nM T64969 C9XIA1 44580891 IC50 = 109 nM T64969 CZC2R9 44580892 IC50 = 130 nM T64969 CYSF35 44580915 IC50 = 120 nM T64969 CP81ZN 44580916 IC50 = 58 nM T64969 CQL7G0 44580917 IC50 = 140 nM T64969 C8LK3H 44580918 IC50 = 14 nM T64969 C5H1XE 44580949 IC50 = 115 nM T64969 C2I8SC 44580950 IC50 = 81 nM T64969 CK9NC7 44580951 IC50 = 63 nM T64969 CO6A7L 44580971 IC50 = 141 nM T64969 CHSR02 44581016 IC50 = 60 nM T64969 C06LHO 44581017 IC50 = 50 nM T64969 CQV6W9 44586019 IC50 = 670 nM T64969 C5WOE2 44586449 IC50 = 300 nM T64969 C0VF8M 44586450 IC50 = 2200 nM T64969 C4K7NP 44586451 IC50 = 3400 nM T64969 C1JNR5 44586452 IC50 = 4700 nM T64969 C6T8UP 44586490 IC50 = 22800 nM T64969 CU95NI 44586526 IC50 > 200000 nM T64969 CBK9R3 44586527 IC50 = 1320 nM T64969 CA18IW 44586528 IC50 = 3180 nM T64969 C0YSZ2 44586577 IC50 > 200000 nM T64969 CTHK89 44587526 IC50 = 49 nM T64969 C7BP3R 44587569 IC50 = 9 nM T64969 CXN7Z2 44592167 IC50 = 82 nM T64969 CM16KD 44592210 IC50 = 7 nM T64969 C6OZB8 44592211 IC50 = 10 nM T64969 C9NXT5 44592212 IC50 = 9 nM T64969 C70GPR 44592213 IC50 = 14 nM T64969 CKC47E 44592253 IC50 = 59 nM T64969 CZW9G8 44592254 IC50 = 17900 nM T64969 CQKV92 44592255 IC50 = 27 nM T64969 C3XAR9 44592374 IC50 = 11 nM T64969 CL2Z5Q 44592375 IC50 = 6 nM T64969 COY57J 44592504 IC50 = 10000 nM T64969 C3M0SR 44593598 IC50 = 0.01 ug.mL-1 T64969 C70VZY 44593599 IC50 = 0.2 ug.mL-1 T64969 C6OC4Z 44607530 IC50 < 0.5 nM T64969 C8M5KI 44611919 IC50 = 68.2 nM T64969 C1EM3P 44629538 IC50 < 1 nM T64969 C2SHM5 44723861 IC50 = 3740 nM T64969 CJ2L1M 44820629 IC50 = 2200 nM T64969 CP2YM3 45103907 IC50 = 2400 nM T64969 C13CJG 45139788 IC50 = 1400 nM T64969 CD78OC 45139973 IC50 = 600 nM T64969 CU3RF1 45139989 IC50 > 10000 nM T64969 CQGZ06 45139991 IC50 > 10000 nM T64969 CXR3J0 45140149 IC50 = 28.8 nM T64969 C42EAO 45140150 IC50 = 1.99 nM T64969 CQ0WZ2 45140151 IC50 = 15.4 nM T64969 CCLE50 45140153 IC50 = 99.4 nM T64969 C4QVP3 45140347 IC50 = 268 nM T64969 CR8GN7 45140348 IC50 = 5077 nM T64969 C6K1JW 45140349 IC50 = 12.8 nM T64969 C82WLQ 45140350 IC50 = 125.6 nM T64969 CR4C9A 45140351 IC50 = 614 nM T64969 CB43GO 45141138 IC50 = 1.24 nM T64969 C61XCE 45141139 IC50 = 9.25 nM T64969 C4TEA9 45141140 IC50 = 291 nM T64969 C7YI9T 45141141 IC50 = 23.6 nM T64969 C47QIR 45141349 IC50 = 0.17 nM T64969 CTDP02 45141350 IC50 = 0.36 nM T64969 CU4RX5 45141351 IC50 = 0.85 nM T64969 C94WSQ 45141352 IC50 = 129 nM T64969 C8I4EW 45141586 IC50 = 0.37 nM T64969 CR4P3U 45151149 IC50 = 7480 nM T64969 C7W3UH 45151160 IC50 = 4680 nM T64969 C8C3JW 45151163 IC50 = 5710 nM T64969 CRM6V8 45151173 IC50 = 5070 nM T64969 CU29PK 45151176 IC50 = 4940 nM T64969 C0O6UA 45151186 IC50 = 7780 nM T64969 C8UGV5 45151203 IC50 = 6920 nM T64969 C6F8UE 45261965 IC50 = 350 nM T64969 C0T2MQ 45262036 IC50 = 4 nM T64969 CO28YF 45262447 IC50 = 20 nM T64969 CC31AL 45262457 IC50 > 100000 nM T64969 C5G9AS 45262479 IC50 = 444 nM T64969 C4DT3N 45262482 IC50 = 11 nM T64969 CC6RQ4 45262483 IC50 = 58 nM T64969 C87GSB 45262544 IC50 = 12.3 nM T64969 CX90FV 45265311 IC50 = 0.47 nM T64969 C2E3BZ 45265326 IC50 = 48 nM T64969 CO76KT 45265373 IC50 = 12.6 nM T64969 C56FXL 45265376 IC50 = 158 nM T64969 C5R3XP 45265596 IC50 = 460 nM T64969 C4DK0O 45265630 IC50 > 10000 nM T64969 CIX15N 45266023 IC50 = 120.23 nM T64969 CI82UE 45270897 IC50 > 10000 nM T64969 CKNP14 45276457 IC50 > 100000 nM T64969 CA4T0D 45276458 IC50 > 100000 nM T64969 C9BQM3 45370166 IC50 = 24 nM T64969 C6E2SC 45482700 IC50 > 10000 nM T64969 CZXH74 45482750 IC50 > 10000 nM T64969 CB6X7D 45483674 IC50 = 23 nM T64969 CCMU48 45483675 IC50 = 23 nM T64969 C9PE3R 45483677 IC50 = 19 nM T64969 CF9SL7 45483685 IC50 = 44 nM T64969 CE7J8I 45483687 IC50 = 30 nM T64969 CULV14 45483689 IC50 = 38 nM T64969 C2V0QA 45483691 IC50 = 40 nM T64969 CFN61Z 45483693 IC50 = 38 nM T64969 CET9K4 45483694 IC50 = 45 nM T64969 CJ1XL4 45483695 IC50 = 21 nM T64969 CO0U2K 45483696 IC50 = 33 nM T64969 CKSM90 45483699 IC50 = 111 nM T64969 C7JH2B 45485483 IC50 = 240 nM T64969 C5QVD7 45485488 IC50 = 180 nM T64969 CN3BQ4 45485489 IC50 = 720 nM T64969 CJ1A3L 45485503 IC50 = 500 nM T64969 CCF08Z 45485522 IC50 = 390 nM T64969 C4HS8N 45485552 IC50 = 770 nM T64969 CB4N0W 46184985 IC50 = 70 nM T64969 C71BUZ 46197015 IC50 < 1 nM T64969 C3HC5D 46197127 IC50 = 16 nM T64969 CZ7W0G 46197128 IC50 = 1.7 nM T64969 CK9Y2G 46197129 IC50 = 30 nM T64969 C5VC7I 46200951 IC50 = 80 nM T64969 C5G7SV 46207008 IC50 = 7820 nM T64969 CA3N9W 46207009 IC50 = 940 nM T64969 C4K9MS 46207010 IC50 = 1720 nM T64969 CAE1M9 46207011 IC50 = 9460 nM T64969 C2F4HI 46207012 IC50 = 11570 nM T64969 C7CID4 46207014 IC50 = 31430 nM T64969 C9CER0 46207015 IC50 > 50000 nM T64969 CPI6S1 46207036 IC50 = 29830 nM T64969 C3F6SM 46207037 IC50 > 50000 nM T64969 C10WUT 46207039 IC50 = 35290 nM T64969 CPXZ65 46207040 IC50 = 22810 nM T64969 C30QNX 46207041 IC50 = 14720 nM T64969 CDN84U 46207042 IC50 = 90 nM T64969 CV1P0R 46207043 IC50 = 17510 nM T64969 C41RBD 46207062 IC50 = 19260 nM T64969 CBQS73 46207441 IC50 = 750 nM T64969 C1WS6M 46207442 IC50 = 1490 nM T64969 CUA97D 46209401 IC50 > 10000 nM T64969 CWN74L 46209503 IC50 = 6900 nM T64969 CKY01V 46209504 IC50 > 10000 nM T64969 CDE1W6 46212905 IC50 = 8 nM T64969 CL41UW 46212970 IC50 = 7 nM T64969 CJR09Y 46212971 IC50 = 0.043 nM T64969 CF57GK 46215462 IC50 = 3900 nM T64969 CY3HW5 46224684 IC50 = 940 nM T64969 C1U7IT 46225595 IC50 = 63 nM T64969 C8YPN0 46225596 IC50 = 350 nM T64969 C34JTS 46225597 EC50 > 10000 nM T64969 CGD73B 46225598 IC50 > 10000 nM T64969 C3E0PU 46225599 IC50 = 4500 nM T64969 CRDY89 46225610 IC50 = 16 nM T64969 C0JMT8 46225611 IC50 = 200 nM T64969 CF0D5J 46225612 IC50 = 46 nM T64969 CFVO38 46225632 IC50 = 2300 nM T64969 CLZ1O6 46225634 IC50 = 805 nM T64969 C07VDX 46225635 IC50 = 670 nM T64969 CT70DX 46225640 IC50 = 32 nM T64969 CJUF68 46225641 IC50 = 44 nM T64969 C6AJ5N 46225647 IC50 = 730 nM T64969 C2WCV1 46225648 IC50 > 10000 nM T64969 CBS96A 46225649 IC50 > 10000 nM T64969 C38BFC 46225657 EC50 = 9400 nM T64969 CD0A6F 46225658 IC50 = 1400 nM T64969 C1B3KS 46225663 IC50 = 430 nM T64969 CU46XI 46225664 IC50 = 260 nM T64969 CO3HS2 46225665 EC50 > 10000 nM T64969 C2UV1S 46225666 EC50 > 10000 nM T64969 CX5B1G 46225667 IC50 = 6200 nM T64969 C2Q9OH 46225668 IC50 = 1400 nM T64969 C16LEO 46225679 IC50 = 2200 nM T64969 CM14FH 46225680 IC50 = 230 nM T64969 CQS96E 46225681 IC50 > 10000 nM T64969 CJIK35 46225682 IC50 = 15 nM T64969 C8S4QA 46225688 IC50 = 250 nM T64969 CYBD14 46229355 IC50 = 1980 nM T64969 C7XEG1 46229356 IC50 = 2240 nM T64969 CO0DJ5 46229377 IC50 = 21710 nM T64969 C5Y1PT 46229378 IC50 = 4150 nM T64969 CE25DB 46229379 IC50 = 4680 nM T64969 CT70VJ 46229380 IC50 = 27350 nM T64969 CT15NR 46229381 IC50 = 960 nM T64969 CG14AQ 46229405 IC50 = 1070 nM T64969 CK7BT5 46229406 IC50 = 7510 nM T64969 CKN40P 46229407 IC50 = 1860 nM T64969 CKL7Z5 46229408 IC50 = 1120 nM T64969 C3IS6A 46229409 IC50 = 9260 nM T64969 CEK82A 46229459 IC50 = 32120 nM T64969 C3N0HQ 46229460 IC50 = 36880 nM T64969 CAO23J 46229461 IC50 > 50000 nM T64969 CJ3FW1 46229462 IC50 > 50000 nM T64969 CI6RL4 46229463 IC50 > 50000 nM T64969 CQ8K2T 46229464 IC50 > 50000 nM T64969 C2SF0M 46229498 IC50 = 670 nM T64969 CY4K7S 46229499 IC50 = 980 nM T64969 C9YBX1 46229500 IC50 = 8540 nM T64969 CF4P3E 46229516 IC50 = 19410 nM T64969 CI1X8G 46229517 IC50 = 120 nM T64969 CH91IA 46229518 IC50 = 3460 nM T64969 CW40RS 46229519 IC50 = 560 nM T64969 CS3OP4 46229535 IC50 = 870 nM T64969 C7UOQ9 46229536 IC50 = 5830 nM T64969 C4MA6T 46229537 IC50 = 18120 nM T64969 CUSX60 46229538 IC50 = 22040 nM T64969 CAKH92 46229539 IC50 = 43210 nM T64969 CLOQ02 46229565 IC50 = 24650 nM T64969 CWD64Q 46229566 IC50 = 31940 nM T64969 CJ4NH6 46229567 IC50 > 50000 nM T64969 C6L0RY 46229767 IC50 = 2.53 nM T64969 CAZ5R0 46229769 IC50 = 87.1 nM T64969 CGMY03 46229773 IC50 = 80 nM T64969 CE12JD 46229813 IC50 = 32.7 nM T64969 CU0RG6 46229815 IC50 > 1000 nM T64969 C31DLC 46229816 IC50 = 32.6 nM T64969 CN2OI5 46229817 IC50 = 106 nM T64969 C5D0OS 46229856 IC50 = 31180 nM T64969 CV96NK 46230527 IC50 = 25.9 nM T64969 C6N7SV 46230529 IC50 = 14.8 nM T64969 C37XZC 46230531 IC50 = 17.7 nM T64969 CYZV41 46231219 IC50 > 8480 nM T64969 C7J5UP 46231220 IC50 = 1688 nM T64969 CC96GZ 46231221 IC50 = 5797 nM T64969 CEOD43 46231624 IC50 = 9120 nM T64969 CXD3E9 46231625 IC50 = 7230 nM T64969 C4J1RQ 46231626 IC50 = 5840 nM T64969 C4XU2C 46231627 IC50 = 4960 nM T64969 CU26ZF 46231684 IC50 = 3110 nM T64969 CA51RN 46231685 IC50 = 1720 nM T64969 CWM8V1 46231686 IC50 = 1010 nM T64969 C2VDX3 46231687 IC50 = 48 nM T64969 CS6I0D 46231742 IC50 = 692 nM T64969 CC0J3D 46231743 IC50 = 1589 nM T64969 CE38ZP 46231744 IC50 = 8710 nM T64969 CTYE12 46231745 IC50 = 6280 nM T64969 C6QG4O 46231746 IC50 = 5330 nM T64969 CE23SX 46231817 IC50 = 3580 nM T64969 CADC90 46231818 IC50 = 2140 nM T64969 C1XV2H 46231819 IC50 = 1270 nM T64969 CLN2B6 46231820 IC50 = 316 nM T64969 CPN4S3 46231883 IC50 = 35 nM T64969 C35LAZ 46231884 IC50 = 464 nM T64969 C5Y3DS 46231885 IC50 = 1350 nM T64969 CYT37A 46232443 IC50 > 50000 nM T64969 C48ZVW 46232555 IC50 > 50000 nM T64969 CS9B1U 46232556 IC50 > 50000 nM T64969 C7ON5A 46233287 IC50 > 10000 nM T64969 CS8P3R 46233390 IC50 = 72 nM T64969 C0QP3Y 46239453 IC50 = 8.59 nM T64969 CZD79U 46831432 IC50 = 12.5 nM T64969 CNWU53 46831433 IC50 = 24.8 nM T64969 C7HK3L 46831434 IC50 = 0.27 nM T64969 CJ9IY2 46831435 IC50 = 0.23 nM T64969 CJ0OF3 46842881 IC50 = 1360 nM T64969 CFP21E 46842882 IC50 = 2170 nM T64969 CN8D3H 46842883 IC50 = 340 nM T64969 CD3TK2 46842884 IC50 = 70 nM T64969 C6UIO0 46842885 IC50 = 130 nM T64969 CGA46B 46842886 IC50 = 3060 nM T64969 CC0I7S 46842887 IC50 = 5190 nM T64969 C9IJ6M 46842888 IC50 = 3870 nM T64969 CBR9Z1 46842916 IC50 = 830 nM T64969 CB2AL1 46842917 IC50 = 4210 nM T64969 CW2BF1 46842918 IC50 = 6270 nM T64969 CIM0F8 46842919 IC50 = 7320 nM T64969 CYTG25 46842920 IC50 = 7780 nM T64969 CUEF65 46842921 IC50 = 11270 nM T64969 CYS9U5 46842922 IC50 = 12260 nM T64969 CDM32Q 46842923 IC50 = 10970 nM T64969 CS3Q7I 46842945 IC50 = 6560 nM T64969 CZ92NO 46842946 IC50 = 7380 nM T64969 C5BGH3 46842947 IC50 = 6850 nM T64969 C9BI7M 46842971 IC50 = 13370 nM T64969 CFR1C6 46845026 IC50 > 300000 nM T64969 CW0P5B 46845702 IC50 = 1060 nM T64969 C7KM0E 46845704 IC50 = 1250 nM T64969 C8ETL6 46854891 IC50 = 82 nM T64969 CKL98B 46854893 IC50 = 452 nM T64969 C0HT9B 46855200 IC50 = 223 nM T64969 C8VX3G 46855360 IC50 = 820 nM T64969 CE3WH9 46865125 IC50 = 4.1 nM T64969 C45LYT 46865445 IC50 = 30.4 nM T64969 CCBE34 46865992 IC50 = 220 nM T64969 C1XEY4 46866615 IC50 = 13.5 nM T64969 CF6K3E 46866616 IC50 = 10.8 nM T64969 CLS29B 46872626 IC50 > 10000 nM T64969 C2MCT8 46879471 IC50 = 867 nM T64969 C6M0JK 46879472 IC50 = 1210 nM T64969 CGV58U 46879473 IC50 > 10000 nM T64969 C8GD2E 46879474 IC50 = 15140 nM T64969 CF4OY7 46881850 IC50 = 58 nM T64969 CEKX49 46881918 IC50 = 58 nM T64969 CMVZ46 46886319 Ki = 31.62 nM T64969 CJR01I 46886321 IC50 = 50 nM T64969 C2O8RZ 46886323 IC50 = 610 nM T64969 CC7MG8 46886325 IC50 = 350 nM T64969 C3T6YO 46886327 IC50 = 1000 nM T64969 CA57MX 46886970 IC50 = 2500 nM T64969 CRGH62 46886971 IC50 = 161600 nM T64969 C68AGR 46886972 IC50 = 27200 nM T64969 CP32GW 46886973 IC50 = 55200 nM T64969 C48JWD 46886974 IC50 = 91700 nM T64969 C7H3MD 46887038 IC50 = 45600 nM T64969 C40NOR 46887039 IC50 = 96400 nM T64969 C7I4SB 46887074 IC50 > 300000 nM T64969 CI5QX2 46887110 IC50 > 300000 nM T64969 C0Q7NG 46887111 IC50 > 300000 nM T64969 CU15AN 46887112 IC50 = 33100 nM T64969 CD90BV 46887113 IC50 > 300000 nM T64969 CH3O9K 46887255 IC50 > 200000 nM T64969 C7NUT3 46887298 IC50 > 200000 nM T64969 CWV65D 46887299 IC50 > 200000 nM T64969 CH5BZ6 46887300 IC50 > 200000 nM T64969 C20UCB 46887348 IC50 > 200000 nM T64969 C0KEG5 46887349 IC50 > 200000 nM T64969 CY59RB 46887397 IC50 = 56100 nM T64969 CL5R0D 46888599 IC50 = 1630 nM T64969 C3IE0X 46888601 IC50 = 980 nM T64969 C1A0XQ 46888603 IC50 = 4400 nM T64969 CB5YQ1 46888635 IC50 = 1920 nM T64969 C6YC4O 46888663 IC50 = 1300 nM T64969 C0AUT8 46888665 IC50 = 2070 nM T64969 CAZT96 46888666 IC50 > 50000 nM T64969 CS4U3P 46888668 IC50 = 2450 nM T64969 CASV10 46888710 IC50 = 1370 nM T64969 CY2TV5 46888712 IC50 = 2750 nM T64969 CX5AL6 46888740 IC50 = 2500 nM T64969 CSWE93 46888742 IC50 = 15120 nM T64969 CW7AR1 46889887 IC50 > 1000 nM T64969 CMNK35 46889911 IC50 > 1000 nM T64969 C0WYM1 46898022 IC50 = 10000 nM T64969 CB92VU 46912443 IC50 > 200000 nM T64969 CU6HC7 46912444 IC50 = 31200 nM T64969 C8A4KU 46912445 IC50 = 1200 nM T64969 CNOS56 46912446 IC50 = 143500 nM T64969 CV38NE 46912546 IC50 = 500 nM T64969 CRI1Q8 46912936 IC50 = 620 nM T64969 C60GAV 46929544 IC50 > 8000 nM T64969 CP34VL 46929748 IC50 > 1000 nM T64969 CJ2E9Q 46929857 IC50 > 25000 nM T64969 C47TGL 46935972 IC50 = 1730 nM T64969 CQVZ79 46935973 IC50 = 2360 nM T64969 CD1N7L 46935974 IC50 = 1840 nM T64969 C7T0ZG 46935975 IC50 = 3850 nM T64969 C12XQO 46936026 IC50 = 2670 nM T64969 C16OAQ 46936027 IC50 = 3080 nM T64969 CBZM62 46936028 IC50 = 1920 nM T64969 C5M0XC 46936029 IC50 = 60 nM T64969 C4H7YB 46936030 IC50 = 190 nM T64969 C19JEL 46936031 IC50 = 370 nM T64969 C6PYR0 46936080 IC50 = 630 nM T64969 CXIN65 46936081 IC50 = 1040 nM T64969 CZ7QW6 46936082 IC50 = 820 nM T64969 CY65UA 46936083 IC50 = 970 nM T64969 CX6A9S 46936084 IC50 = 11240 nM T64969 C4FJA3 46936085 IC50 = 9370 nM T64969 CCUW64 46936126 IC50 = 8950 nM T64969 CS4I3P 46936127 IC50 = 15720 nM T64969 CRKD93 46936128 IC50 = 19640 nM T64969 CR9D8U 46936129 IC50 = 10170 nM T64969 CCHU82 46936130 IC50 = 22360 nM T64969 CE70ZG 46936131 IC50 = 24160 nM T64969 C0IDM5 46936170 IC50 = 17840 nM T64969 C67CSG 46936171 IC50 = 25740 nM T64969 C08QUC 46936172 IC50 = 24370 nM T64969 C9WRB7 46936173 IC50 = 28170 nM T64969 CJ0ZY8 46936174 IC50 = 19830 nM T64969 C60DLE 46936175 IC50 = 21520 nM T64969 CUT3S0 46937464 IC50 = 1.81 nM T64969 C41JQX 46937466 IC50 = 23.02 nM T64969 C2QRW8 46937467 IC50 = 0.57 nM T64969 CONM83 46937468 IC50 = 4.05 nM T64969 C4PZ8J 46937511 IC50 = 0.22 nM T64969 CK5U2C 46937558 IC50 = 0.22 nM T64969 CBZX50 46937560 IC50 = 0.22 nM T64969 C43QHB 46937562 IC50 = 0.22 nM T64969 CBR76Q 46937566 IC50 = 0.22 nM T64969 CPR6O9 47108694 IC50 = 11910 nM T64969 CM24GY 47108695 IC50 = 6740 nM T64969 CF9ZH7 47108713 IC50 = 17810 nM T64969 C4SF5L 47108741 IC50 = 90 nM T64969 CCYJ10 47108773 IC50 = 2080 nM T64969 CJ4T3N 47120995 IC50 = 590 nM T64969 CJS49Y 47232283 IC50 = 3270 nM T64969 CE4SU5 47298428 IC50 > 10000 nM T64969 CCWB05 49788361 IC50 = 720 nM T64969 C0J6HA 49788362 IC50 > 20000 nM T64969 C1OLV6 49788363 IC50 = 1270 nM T64969 CLH4N7 49788364 IC50 = 91 nM T64969 CG0YF3 49788365 IC50 = 3057 nM T64969 COWP56 49788366 IC50 = 20 nM T64969 C93ROW 49788425 IC50 = 46 nM T64969 CM8X1I 49788426 IC50 = 3503 nM T64969 C8XN1P 49788427 IC50 = 9 nM T64969 C3PM9Q 49788428 IC50 = 21 nM T64969 C8AS0L 49788429 IC50 = 89 nM T64969 C31VOW 49788430 IC50 > 20000 nM T64969 C5MZY4 49788490 IC50 = 12 nM T64969 CFLD56 49788491 IC50 = 12 nM T64969 CTQ5M0 49788492 IC50 = 149 nM T64969 CU6Y9D 49788493 IC50 = 4884 nM T64969 C2TY0A 49788560 IC50 > 20000 nM T64969 CE2ST8 49788561 IC50 = 1090 nM T64969 C0EK8U 49788642 IC50 > 20000 nM T64969 CV6O3H 49798025 IC50 = 85 nM T64969 C4FJ0Y 49798860 IC50 = 3880 nM T64969 CBX8W0 49798861 IC50 = 5760 nM T64969 CRLT80 49798983 IC50 = 24150 nM T64969 CL5ZR3 49798984 IC50 = 25470 nM T64969 C26DKM 49798985 IC50 = 15560 nM T64969 CQ80WE 49799021 IC50 = 20610 nM T64969 CX19VP 49799195 IC50 = 8920 nM T64969 CJYK69 49799238 IC50 = 6430 nM T64969 C7NV4K 49799239 IC50 = 7280 nM T64969 C8AWO3 49799240 IC50 = 5270 nM T64969 C37BOI 49799285 IC50 = 17490 nM T64969 CL57XI 49799286 IC50 = 15240 nM T64969 CG3FX1 49799287 IC50 = 21480 nM T64969 C1UPR7 49799323 IC50 = 17310 nM T64969 CO3G7R 49799361 IC50 = 18450 nM T64969 CET2D6 49799362 IC50 = 19320 nM T64969 C05PNX 49799381 IC50 = 16140 nM T64969 CC2WR7 49799382 IC50 = 18350 nM T64969 C7DS9L 49799452 IC50 = 5740 nM T64969 C4B0VH 49799526 IC50 = 10640 nM T64969 CY46VG 49799527 IC50 = 8090 nM T64969 CA26HX 49799528 IC50 = 9830 nM T64969 C69YEO 49799573 IC50 = 10060 nM T64969 CM6HD2 49799574 IC50 = 8150 nM T64969 COD7X8 49799764 IC50 = 3240 nM T64969 C3PNH8 49799765 IC50 = 8110 nM T64969 CO89EH 49799766 IC50 = 10850 nM T64969 C4MYV3 49799767 IC50 = 6820 nM T64969 CK92JP 49799768 IC50 = 1270 nM T64969 CY32VC 49799770 IC50 = 25000 nM T64969 C21GOI 49799777 IC50 = 4120 nM T64969 C7QR3M 49799778 IC50 = 3620 nM T64969 CVEG83 49799781 IC50 = 26740 nM T64969 C6X5MK 49799782 IC50 = 20810 nM T64969 C2GXI7 49799783 IC50 = 24320 nM T64969 C1NI4A 49799785 IC50 = 32000 nM T64969 C3VQ9Z 49799786 IC50 = 14530 nM T64969 CAL42P 49799787 IC50 = 12420 nM T64969 C49XCZ 49799788 IC50 = 13870 nM T64969 CHSF07 49806372 IC50 > 1000 nM T64969 C5ME3S 49806721 IC50 > 50000 nM T64969 C3ZI9B 49840051 IC50 > 10000 nM T64969 CDFE41 49840052 IC50 > 10000 nM T64969 C1XHO0 49840114 IC50 > 10000 nM T64969 CIMT03 49840186 IC50 > 10000 nM T64969 CIX4E3 49840245 IC50 > 10000 nM T64969 CLWN26 49840246 IC50 > 10000 nM T64969 CN89TG 49840317 IC50 > 10000 nM T64969 C0AJ9R 49840318 IC50 > 10000 nM T64969 CF91RS 49843531 IC50 > 10000 nM T64969 CE7D2J 49855568 IC50 = 2.5 nM T64969 CFD9P3 49855569 IC50 = 4.8 nM T64969 C1AU5N 49855758 IC50 = 18 nM T64969 CIFK93 49855759 IC50 = 2.9 nM T64969 CK48OJ 49855760 IC50 = 2.8 nM T64969 CZI3M1 49855761 IC50 = 26 nM T64969 CRPZ58 49855949 IC50 = 49 nM T64969 CTU0K3 49855950 IC50 = 29 nM T64969 CF85NL 49855951 IC50 = 15 nM T64969 CF7YS9 49855952 IC50 = 3.9 nM T64969 CJU38G 49855953 IC50 = 2.2 nM T64969 C9Z8ED 49859891 IC50 = 1000 nM T64969 CB5O0I 49860186 IC50 = 200 nM T64969 C9W6SO 49860190 IC50 = 90 nM T64969 CF4V7Z 49867019 IC50 = 2200 nM T64969 C5RQ7C 50908680 Ki = 500 nM T64969 CD2K4R 50908681 Ki = 400 nM T64969 C6XYT1 50941838 IC50 > 100000 nM T64969 C61DVY 50990961 IC50 = 4900 nM T64969 CV3UP9 50992247 IC50 = 190 nM T64969 CS9G6E 50997096 IC50 > 10000 nM T64969 CM42BY 51000510 Ki = 296000 nM T64969 CAZQ43 51003133 IC50 > 1000 nM T64969 CDU4Q5 51346827 Ki > 1800 nM T64969 C49ZVC 51346878 IC50 = 240 nM T64969 CJ4L1K 51346887 IC50 = 120 nM T64969 CH1TU2 51346888 IC50 = 3 nM T64969 CH1WR3 52914084 IC50 = 149 nM T64969 C13MUQ 52914647 IC50 = 281 nM T64969 CXA03W 52920796 IC50 > 100 nM T64969 CEQN27 52936621 Ki > 1000 nM T64969 CM24LF 52938983 IC50 = 101.4 nM T64969 CAD1N6 52940774 IC50 = 0.03 nM T64969 CU1P2L 52940797 IC50 = 8010 nM T64969 C4R7IM 52941368 IC50 = 253600 nM T64969 C2ZTN3 52941514 IC50 = 2880 nM T64969 CDHJ08 52942235 IC50 = 100000 nM T64969 CG9E4A 52942446 Ki > 1000000 nM T64969 C8SJ2Q 52942862 Ki > 1000000 nM T64969 C7BY6M 52942956 IC50 = 111400 nM T64969 CT8VW3 52943139 IC50 > 10000 nM T64969 C1XEV2 52943394 IC50 = 20500 nM T64969 CA62KU 52944152 IC50 = 160300 nM T64969 CLO46D 52944812 Ki = 3450 nM T64969 CWPC54 52945348 IC50 = 638 nM T64969 CQV34K 52945403 IC50 > 200000 nM T64969 C4NLX7 52945630 IC50 = 54200 nM T64969 CXD6T8 52945845 IC50 = 2800 nM T64969 CQ87LD 52946569 IC50 = 78 nM T64969 C97XZA 52946619 IC50 > 200000 nM T64969 C8QNI5 52946868 IC50 = 8.12 nM T64969 C2WM9K 52947210 IC50 = 5900 nM T64969 CE0X5U 52947574 IC50 > 200000 nM T64969 CD9S4I 52947801 IC50 = 529300 nM T64969 CA6IL3 52947802 IC50 > 200000 nM T64969 CI6GX2 52948511 Ki = 680 nM T64969 C2KAJ4 52948634 IC50 = 53100 nM T64969 CWA74O 52949707 Ki = 590 nM T64969 C0A1GQ 52949915 IC50 = 12800 nM T64969 C6OTY5 53251320 IC50 > 30000 nM T64969 C09SDH 53257410 IC50 > 10000 nM T64969 CX13OD 53316491 IC50 = 150 nM T64969 CJ61BU 53317172 IC50 > 100000 nM T64969 C89QOE 53317173 IC50 = 17 nM T64969 C50BWT 53317174 IC50 = 590 nM T64969 C39KUD 53317175 IC50 = 38 nM T64969 C1NLD5 53317828 IC50 = 4100 nM T64969 CE8OY2 53317913 IC50 > 100 nM T64969 CBHT02 53318117 IC50 = 950 nM T64969 CX1V9L 53318118 IC50 = 670 nM T64969 C90MNQ 53318457 IC50 = 1100 nM T64969 C2X8OF 53318458 IC50 = 18 nM T64969 CK59QY 53318459 IC50 = 270 nM T64969 CZS8K4 53319042 Ki > 1800 nM T64969 C3MUN7 53319130 IC50 = 2200 nM T64969 C1PMT2 53319131 IC50 = 55600 nM T64969 CRBE56 53319790 IC50 = 34 nM T64969 CSC61X 53320059 IC50 = 114 nM T64969 CUD21V 53320263 Ki > 1800 nM T64969 C4QU3S 53320463 IC50 = 6900 nM T64969 CX65KS 53321087 IC50 = 10000 nM T64969 C3G2WX 53321754 IC50 = 28000 nM T64969 CX7S8I 53322057 IC50 > 1000 nM T64969 CSY76U 53322058 IC50 = 210 nM T64969 C7Y3ZR 53322413 IC50 = 640 nM T64969 CR12OB 53322414 IC50 = 156 nM T64969 CR4K7J 53322690 IC50 = 65 nM T64969 CESA85 53323614 Ki > 1800 nM T64969 CT1BN7 53324027 IC50 = 47000 nM T64969 C43BZJ 53324200 IC50 = 20000 nM T64969 CI6A9B 53324357 IC50 = 1300 nM T64969 CB80KQ 53324440 IC50 = 12800 nM T64969 CGL6Y7 53324441 IC50 = 45200 nM T64969 CG18XC 53325046 IC50 = 1200 nM T64969 CD91UQ 53325047 IC50 = 22000 nM T64969 C5C1UW 53325048 IC50 = 68 nM T64969 CRT07X 53325049 IC50 = 28 nM T64969 C69AUF 53325050 IC50 = 11 nM T64969 CN1X9I 53325551 IC50 = 19 nM T64969 C36OQR 53325588 IC50 > 1000 nM T64969 CNX76J 53325743 IC50 = 20800 nM T64969 C07PMQ 53326342 IC50 = 4130 nM T64969 CD86WI 53328229 IC50 = 4 nM T64969 C5ETO8 53328965 IC50 = 3 nM T64969 CCZG21 53328969 IC50 = 1600 nM T64969 CJ2Y5P 53330551 IC50 = 13 nM T64969 CNPM14 53341082 IC50 = 3.3 nM T64969 C0SWH5 53348216 IC50 > 40000 nM T64969 C8ZRE3 53356518 IC50 > 16670 nM T64969 CM7P3W 53357328 IC50 > 50000 nM T64969 C4PO3Z 53357348 IC50 = 1929 nM T64969 CXW05L 53357349 IC50 = 12070 nM T64969 CBK9Q6 53357848 IC50 > 10000 nM T64969 C8NA4L 53384644 IC50 > 30000 nM T64969 CVG90B 53389651 IC50 > 10000 nM T64969 CA50GN 53466759 IC50 < 7 nM T64969 CJ1NB9 53484041 IC50 = 940 nM T64969 CREZ21 53484042 IC50 = 120 nM T64969 C0HN6L 53484043 IC50 = 190 nM T64969 C8D9XG 53736592 IC50 > 10000 nM T64969 C9MBJ6 53759588 IC50 = 4.7 nM T64969 CH53KW 54576742 IC50 = 350 nM T64969 CK1EM6 54580365 IC50 > 10000 nM T64969 C4SN3X 54580366 IC50 > 10000 nM T64969 CQ9I1X 54580996 IC50 = 67 nM T64969 C1HZ4Y 54581368 IC50 > 10000 nM T64969 CA6H2U 54581369 IC50 > 10000 nM T64969 C5P9BQ 54581370 IC50 > 10000 nM T64969 CW7NH3 54582387 IC50 > 10000 nM T64969 C7R4UG 54582388 IC50 > 10000 nM T64969 C9SZ2I 54582389 IC50 > 10000 nM T64969 CL40KE 54583375 IC50 > 10000 nM T64969 C2MFX7 54585296 IC50 > 10000 nM T64969 CY4RH6 54586238 IC50 > 10000 nM T64969 C8QA0M 54586239 IC50 > 10000 nM T64969 C6RX7G 54586507 IC50 = 95 nM T64969 CL1I5C 54587267 IC50 > 10000 nM T64969 C0JMY7 54673975 IC50 = 82900 nM T64969 CUT84L 54678831 IC50 > 100000 nM T64969 CZH60Y 54708982 IC50 = 76400 nM T64969 CUZH35 54754343 IC50 = 390 nM T64969 C1XS2J 54760383 IC50 = 4 nM T64969 C75YDA 54768720 IC50 = 2080 nM T64969 C65TFD 54768721 IC50 = 10950 nM T64969 C1WVC6 54768722 IC50 = 19120 nM T64969 C05SPN 54768723 IC50 = 20480 nM T64969 CRL5O0 54768724 IC50 = 26560 nM T64969 CBN0C3 54768725 IC50 = 17390 nM T64969 CR98HI 54768726 IC50 = 14830 nM T64969 C7B8XU 54768951 IC50 = 1570 nM T64969 CT1P3J 54768952 IC50 = 5110 nM T64969 CMN8T0 54768953 IC50 = 700 nM T64969 CZEC06 54768954 IC50 = 2380 nM T64969 C21KRM 54768955 IC50 = 12240 nM T64969 CJ0Q4M 54768956 IC50 = 8660 nM T64969 CY7B5N 54768957 IC50 = 590 nM T64969 CJAN-67 54768958 IC50 = 9780 nM T64969 CE0O9W 54769185 IC50 = 2170 nM T64969 C8LI9H 54769186 IC50 = 7830 nM T64969 CZE0I1 54769187 IC50 = 410 nM T64969 CE8WK1 54772084 IC50 = 22360 nM T64969 CPMZ93 54772085 IC50 = 23270 nM T64969 CKA7U0 54772086 IC50 = 26000 nM T64969 CC4FN9 54772087 IC50 = 33000 nM T64969 CU8YW6 56325569 IC50 = 45000 nM T64969 CQ17GA 56640518 IC50 = 34.8 nM T64969 CG20VK 56640520 IC50 = 6.8 nM T64969 CZ9C8M 56640588 IC50 = 14.7 nM T64969 CH0D7P 56640590 IC50 = 17.6 nM T64969 CN9QD7 56643097 IC50 > 10000 nM T64969 CK2F5X 56649610 IC50 = 66100 nM T64969 CTF90E 56649640 IC50 = 6.6 nM T64969 CU76CR 56649641 IC50 = 3.8 nM T64969 C1LQT6 56649642 IC50 = 3.3 nM T64969 CT6G3J 56649645 IC50 > 100000 nM T64969 C5D4EP 56659276 IC50 = 60 nM T64969 CPZ62X 56659321 IC50 = 6020 nM T64969 C9XCI1 56659322 IC50 = 1020 nM T64969 CR6VD1 56659589 IC50 = 251.19 nM T64969 C2PYI1 56659875 IC50 = 11290 nM T64969 CT5NK2 56659876 IC50 = 18350 nM T64969 C2MW9D 56659883 IC50 = 21280 nM T64969 CX28ME 56660000 IC50 > 10000 nM T64969 CYZ6C5 56661789 IC50 = 8630 nM T64969 CD0UZ8 56662784 IC50 = 3610 nM T64969 CNE6P1 56662786 IC50 = 2810 nM T64969 CD67RU 56663333 IC50 = 13730 nM T64969 CCR3V9 56663334 IC50 = 24150 nM T64969 C6QY0W 56665233 IC50 = 5560 nM T64969 C7NF0U 56666765 IC50 = 2940 nM T64969 C9LPB6 56666766 IC50 = 21840 nM T64969 C4S9ID 56666767 IC50 = 32850 nM T64969 CT3BC2 56669670 IC50 = 8800 nM T64969 C4L2QB 56670196 IC50 = 3430 nM T64969 CIPW74 56670197 IC50 = 1510 nM T64969 CSNH68 56670198 IC50 = 15920 nM T64969 C97LHS 56670199 IC50 = 17260 nM T64969 C6W7BR 56670200 IC50 = 38520 nM T64969 CK2B0C 56672168 IC50 = 6310 nM T64969 CS45AF 56673177 IC50 = 3490 nM T64969 CRXF95 56673721 IC50 = 5930 nM T64969 CG9N7C 56673722 IC50 = 6410 nM T64969 CFAT97 56673723 IC50 = 26200 nM T64969 CT85LD 56676436 IC50 = 1210 nM T64969 CL2DT3 56676437 IC50 = 4280 nM T64969 CMO70N 56676438 IC50 = 7220 nM T64969 CXP5G4 56677027 IC50 = 14530 nM T64969 CE40HN 56678885 IC50 = 8430 nM T64969 C6ME8I 56680356 IC50 = 2170 nM T64969 CNLI27 56680357 IC50 = 8280 nM T64969 CN28KJ 56680358 IC50 = 9590 nM T64969 CYT34H 56682199 IC50 = 5350 nM T64969 C21SXU 56682201 IC50 = 7660 nM T64969 CV3QB9 56683074 IC50 = 7710 nM T64969 CX2MU1 56683151 IC50 = 5160 nM T64969 CG6JP0 56683152 IC50 = 6630 nM T64969 CC2E5V 56683153 IC50 = 3450 nM T64969 COK71Z 56683687 IC50 = 5170 nM T64969 CQ8Z1X 56683695 IC50 = 24680 nM T64969 C5GM0Z 56683696 IC50 = 26170 nM T64969 CNL0A1 56683697 IC50 = 18720 nM T64969 CP7M1A 56683698 IC50 = 24330 nM T64969 C12XMC 56735038 IC50 = 38320 nM T64969 CR50TJ 56835147 IC50 > 10000 nM T64969 CI5ZJ7 56835161 IC50 = 190 nM T64969 CVA8U4 56837416 IC50 = 870 nM T64969 C3QD4K 56839586 IC50 = 16.6 nM T64969 CLSN24 56839587 IC50 = 5.54 nM T64969 CW06VF 56839588 IC50 = 24 nM T64969 CRYP21 56839589 IC50 = 5.93 nM T64969 CJRC62 56849701 IC50 = 34 nM T64969 CG5O8V 56933480 IC50 = 47900 nM T64969 C4P2LY 56934730 IC50 = 63 nM T64969 C63NMS 56934846 IC50 = 33 nM T64969 CP9OF7 56934847 IC50 = 27 nM T64969 CP97GH 56934848 IC50 = 29 nM T64969 CGLB90 56934849 IC50 = 14 nM T64969 C8KV0I 56934851 IC50 = 62 nM T64969 CFK7L9 56934853 IC50 = 450 nM T64969 CXN79H 56934855 IC50 = 4608 nM T64969 C42EHX 56934976 IC50 = 8 nM T64969 CXC51G 56934978 IC50 = 17 nM T64969 COM4F5 56934980 IC50 = 9 nM T64969 C54DNK 56934982 IC50 = 95 nM T64969 C1N4LK 56934984 IC50 = 26 nM T64969 C8O0IR 56934986 IC50 = 52 nM T64969 CBO20L 56934988 IC50 = 45 nM T64969 C2XED0 56935104 IC50 = 4 nM T64969 C8JZC2 56935107 IC50 = 1008 nM T64969 CGV1M9 56935337 IC50 = 93300 nM T64969 CAW57M 56935338 IC50 > 100000 nM T64969 C76EOA 56935464 IC50 > 100000 nM T64969 CO62XN 56935468 IC50 > 100000 nM T64969 CQ2U4F 56949987 IC50 = 37 nM T64969 C86USY 56950114 IC50 = 61 nM T64969 CCTI03 56950115 IC50 = 48 nM T64969 C5K3PV 56950116 IC50 = 65 nM T64969 C7U9SL 56951304 IC50 > 50000 nM T64969 C0GQ9I 56951305 IC50 = 112100 nM T64969 C5YT6A 56951306 IC50 = 12620 nM T64969 CB03EH 56951307 IC50 > 200000 nM T64969 CRJ6H8 56953639 IC50 > 10000 nM T64969 C3D6YR 56953640 IC50 > 10000 nM T64969 CZ9F6B 56953642 IC50 > 10000 nM T64969 CTDR35 56953644 IC50 > 10000 nM T64969 CYF6D8 56953645 IC50 = 9800 nM T64969 CR20WU 56953646 IC50 = 9150 nM T64969 C86GAQ 56953648 IC50 > 10000 nM T64969 CMRB39 56953766 IC50 > 10000 nM T64969 CNG63B 56953767 IC50 > 10000 nM T64969 C1OC9P 56953892 IC50 > 10000 nM T64969 CF5AV8 56953893 IC50 > 10000 nM T64969 CBHG03 56953894 IC50 > 10000 nM T64969 CB5I7C 56953895 IC50 = 7050 nM T64969 C1NIS7 56954003 IC50 = 800 nM T64969 CEKO58 56954004 IC50 = 4800 nM T64969 C7FP1R 56954005 IC50 = 6150 nM T64969 C0PY2A 56954006 IC50 = 1000 nM T64969 CU1QF7 56954007 IC50 = 1000 nM T64969 CG9X1J 56954008 IC50 = 6400 nM T64969 CM9Z4I 56954009 IC50 = 4000 nM T64969 CX1U4G 56954130 IC50 = 900 nM T64969 CG1VI6 56954131 IC50 = 900 nM T64969 CLR6J2 56954132 IC50 = 7600 nM T64969 C9OZ7N 56954133 IC50 = 5800 nM T64969 CLJC74 56954134 IC50 = 900 nM T64969 CEWB79 56954135 IC50 = 7200 nM T64969 CY2GE9 56954136 IC50 = 5000 nM T64969 C5ATX6 56954232 IC50 > 10000 nM T64969 CU3T6F 56954234 IC50 > 10000 nM T64969 CMWK36 56954235 IC50 = 9900 nM T64969 CM9O5W 56954236 IC50 > 10000 nM T64969 C35JTA 56954323 IC50 = 9450 nM T64969 CI5MT0 56954324 IC50 > 10000 nM T64969 C06IDB 56954325 IC50 > 10000 nM T64969 CMT80I 56954326 IC50 > 10000 nM T64969 CE68LB 56954327 IC50 > 10000 nM T64969 CA43UF 56954328 IC50 > 10000 nM T64969 CC85JQ 56954429 IC50 = 9100 nM T64969 CP58NG 56954518 IC50 > 10000 nM T64969 C7K1CZ 56954519 IC50 > 10000 nM T64969 CH1X3R 56954520 IC50 > 10000 nM T64969 CMS50D 56954621 IC50 > 10000 nM T64969 C30ALB 56954622 IC50 > 10000 nM T64969 CZN89G 56954623 IC50 > 10000 nM T64969 CI7U1E 56954736 IC50 > 10000 nM T64969 C18BFU 56954737 IC50 > 10000 nM T64969 CO7D3X 56954739 IC50 > 10000 nM T64969 CRZ0M5 56954836 IC50 = 7050 nM T64969 C04JZF 56954837 IC50 = 800 nM T64969 CH98NL 56954839 IC50 = 6150 nM T64969 CN06PL 56954840 IC50 = 1000 nM T64969 CH0SG3 56954841 IC50 = 1000 nM T64969 C3MYG6 56954954 IC50 = 6400 nM T64969 C6WAD7 56954955 IC50 = 4000 nM T64969 CZ82IH 56954956 IC50 = 900 nM T64969 CSBQ86 56954957 IC50 = 900 nM T64969 CIM60L 56954958 IC50 = 7600 nM T64969 C1LC4G 56955061 IC50 = 900 nM T64969 C4OY1T 56955062 IC50 = 7200 nM T64969 CSJ6L7 56955063 IC50 = 5000 nM T64969 C1GA2O 56955275 IC50 > 10000 nM T64969 CT1KX9 56955277 IC50 > 10000 nM T64969 CAK91L 56955954 IC50 = 739 nM T64969 CJ47MX 56963907 IC50 > 10000 nM T64969 C9L6FD 56963908 IC50 > 10000 nM T64969 CE50IB 56963909 IC50 > 10000 nM T64969 CIX32Y 56965877 IC50 = 2820 nM T64969 COXM57 56970372 IC50 = 1510 nM T64969 CPHX64 57325478 IC50 > 50000 nM T64969 CQ9BW4 57325479 IC50 > 50000 nM T64969 CJ0A7O 57336240 IC50 = 7 nM T64969 CW2G7E 57341100 IC50 = 1.47 nM T64969 CF0RI1 57341101 IC50 = 3.52 nM T64969 CE7ID2 57341102 IC50 = 6.95 nM T64969 C5U4EK 57341103 IC50 = 929 nM T64969 CJ14YA 57341104 IC50 = 0.43 nM T64969 C7VX2L 57341295 IC50 = 0.41 nM T64969 C5UC3L 57341296 IC50 = 4.41 nM T64969 CJY51G 57341297 IC50 = 8.81 nM T64969 CTA57G 57341298 IC50 = 1.95 nM T64969 CW7H2P 57341299 IC50 > 1000 nM T64969 CQ0D5S 57341488 IC50 = 0.38 nM T64969 C2L0VD 57341489 IC50 = 0.58 nM T64969 C7WU1S 57341490 IC50 = 0.3 nM T64969 CX01VB 57341491 IC50 = 0.8 nM T64969 C8C4DZ 57341660 IC50 = 0.29 nM T64969 CQR64D 57341661 IC50 = 1.41 nM T64969 CS4YT2 57341662 IC50 = 1.52 nM T64969 CVG52R 57341663 IC50 = 1.67 nM T64969 CFDQ12 57341838 IC50 > 1000 nM T64969 CT53HQ 57341839 IC50 > 1000 nM T64969 CBJW71 57343703 IC50 = 1.16 nM T64969 C34OGM 57343704 IC50 = 4.99 nM T64969 CB0DY1 57343705 IC50 = 29.5 nM T64969 CW7B3X 57343706 IC50 = 16.4 nM T64969 CVD3B0 57381322 IC50 = 65 nM T64969 C2JD7G 57381323 IC50 = 31 nM T64969 CD65MT 57381324 IC50 = 15 nM T64969 C4YFJ5 57384105 IC50 > 200000 nM T64969 CV9RW5 57384106 IC50 > 200000 nM T64969 C8O4DU 57390197 IC50 = 473 nM T64969 C0E5UQ 57390198 IC50 = 108 nM T64969 CLB4Q9 57390199 IC50 = 129 nM T64969 C04YLM 57390200 IC50 > 10000 nM T64969 CT6GK0 57390220 IC50 > 100000 nM T64969 COC5Y3 57390776 IC50 = 9 nM T64969 C20OVM 57390777 IC50 = 24 nM T64969 CNB25Q 57390936 IC50 = 15680 nM T64969 CR4T2Y 57391283 IC50 > 200000 nM T64969 C80RNH 57391987 IC50 = 1671 nM T64969 C8U9EO 57391988 IC50 = 627 nM T64969 CXL95C 57392008 IC50 > 100000 nM T64969 CK04XQ 57392009 IC50 > 100000 nM T64969 CBL74E 57392425 IC50 > 200000 nM T64969 CHS82P 57392588 IC50 = 7 nM T64969 CZBJ71 57392589 IC50 = 79 nM T64969 CH12GK 57392590 IC50 = 74 nM T64969 CY2XK0 57392591 IC50 = 94 nM T64969 CC2AF6 57392917 IC50 = 25360 nM T64969 CTB8R9 57394107 IC50 = 821 nM T64969 CLY6T8 57394393 IC50 > 30000 nM T64969 CH1U8Y 57394394 IC50 = 2640 nM T64969 CE1A9V 57394653 IC50 = 1.4 nM T64969 CNV76Z 57394656 IC50 = 3.35 nM T64969 CG18LI 57394786 IC50 > 200000 nM T64969 CEDP89 57394787 IC50 > 200000 nM T64969 CP6W4C 57394879 IC50 = 166400 nM T64969 CVR13L 57394880 IC50 = 99900 nM T64969 C8W6IG 57395117 IC50 > 30000 nM T64969 CJC5N7 57395350 IC50 = 18.5 nM T64969 CN7S2K 57395407 IC50 = 1640 nM T64969 C9NA7R 57395419 IC50 = 1870 nM T64969 C9CO0F 57395424 IC50 > 10000 nM T64969 CA4Q3Y 57395925 IC50 = 112700 nM T64969 CM18WP 57396070 IC50 = 86 nM T64969 C2HT3R 57396157 IC50 > 30000 nM T64969 CVA2E1 57396158 IC50 = 21560 nM T64969 CGE48O 57396218 IC50 = 27050 nM T64969 CX1S8R 57396219 IC50 = 28660 nM T64969 CUGP85 57396545 IC50 > 200000 nM T64969 CBUP96 57396646 IC50 = 113300 nM T64969 CI3JB2 57396795 IC50 > 100000 nM T64969 CA02UC 57397177 IC50 = 43.7 nM T64969 CSKH73 57397251 IC50 = 3220 nM T64969 CSAZ51 57397252 IC50 = 11220 nM T64969 C0GSP4 57397265 IC50 = 4410 nM T64969 C6NC2K 57397269 IC50 = 370 nM T64969 CWX47O 57397293 IC50 > 100000 nM T64969 C87OHQ 57397677 IC50 > 10000 nM T64969 CO24DL 57397871 IC50 = 22 nM T64969 C5D1MK 57397872 IC50 = 30 nM T64969 CI6UJ0 57397973 IC50 = 29070 nM T64969 C58KTL 57397974 IC50 = 18150 nM T64969 C18HFC 57397975 IC50 = 15020 nM T64969 CNLS72 57398015 IC50 = 19830 nM T64969 CXJ68F 57398331 IC50 > 200000 nM T64969 C14ANY 57398417 IC50 = 69200 nM T64969 CGV35E 57398558 IC50 > 100000 nM T64969 C73MUW 57398687 IC50 = 422 nM T64969 C9RA2M 57398688 IC50 = 342 nM T64969 C8EB1H 57398880 IC50 = 18.7 nM T64969 CNA4C0 57398939 IC50 = 3130 nM T64969 C7ZI0C 57398942 IC50 = 3540 nM T64969 CG9E5X 57399346 IC50 = 523 nM T64969 C9U2ZS 57399744 IC50 = 12 nM T64969 C2GJQ6 57399859 IC50 > 30000 nM T64969 CDF35C 57400360 IC50 = 9021 nM T64969 C8ZYQ6 57400361 IC50 = 9284 nM T64969 CO34ZJ 57400426 IC50 = 55 nM T64969 CH1A8D 57400659 IC50 = 13880 nM T64969 CC3U6B 57400808 IC50 > 40000 nM T64969 CQ5MB9 57401285 IC50 = 650 nM T64969 CMP96A 57401286 IC50 = 98 nM T64969 C0WFY5 57401428 IC50 > 30000 nM T64969 CTX6K2 57401429 IC50 > 30000 nM T64969 CV1K0D 57401637 IC50 > 30000 nM T64969 C9MAH3 57402380 IC50 = 10.8 nM T64969 C9ZKD5 57402437 IC50 = 5670 nM T64969 CKVJ46 57402440 IC50 = 1204 nM T64969 CP2UN4 57402469 IC50 = 29500 nM T64969 CD0W6U 57402866 IC50 = 721 nM T64969 C1B7RI 57403128 IC50 = 1190 nM T64969 CKFJ31 57403923 IC50 = 623 nM T64969 CZSM95 57412684 IC50 > 10000 nM T64969 CT7M3G 57413593 IC50 = 5.5 nM T64969 CM9OF3 57413596 IC50 = 7 nM T64969 C1RS3Y 57415414 IC50 = 7.8 nM T64969 C80BOQ 57415415 IC50 = 510 nM T64969 CSV93M 57415416 IC50 = 960 nM T64969 C3H6UJ 57415417 IC50 = 2300 nM T64969 CW5IS7 57415418 IC50 = 890 nM T64969 C1DS4B 57415535 IC50 = 21 nM T64969 C0W8LA 57415536 IC50 = 2.8 nM T64969 CRB83E 57415537 IC50 = 36 nM T64969 CN53XW 57428969 IC50 = 283.1 nM T64969 CI5U3G 57496699 IC50 = 11 nM T64969 CZ35GD 57496700 IC50 = 33 nM T64969 C4T7PW 57523998 IC50 > 10000 nM T64969 C1Q7LS 57523999 IC50 = 82 nM T64969 CPS79I 57524088 IC50 = 2350 nM T64969 C0CJ8Z 57524184 IC50 = 3315 nM T64969 C8ICV2 57524400 IC50 = 99 nM T64969 CL72NQ 57524403 IC50 = 165 nM T64969 CAU0K1 57524478 IC50 = 188 nM T64969 CWVJ06 57597166 IC50 = 15 nM T64969 CVS51B 57597223 IC50 = 53 nM T64969 C0QUZ4 57597316 IC50 = 47 nM T64969 CD0M7X 57597387 IC50 = 18 nM T64969 CVK0G4 58056356 IC50 > 50000 nM T64969 C4V7FY 58191950 IC50 = 1300 nM T64969 CPCA29 58191961 IC50 = 1200 nM T64969 C7HF1L 58191965 IC50 = 78 nM T64969 C8LWY9 58191997 IC50 = 33 nM T64969 C3VI7D 58229394 IC50 = 650 nM T64969 CNXU29 58229412 IC50 = 1128 nM T64969 C52OMW 58229434 IC50 = 592 nM T64969 C6BPR2 58985201 IC50 > 50000 nM T64969 C40EXM 59151065 IC50 < 1 nM T64969 C1SI3L 59174579 IC50 = 737 nM T64969 CXN56R 59174683 IC50 = 500 nM T64969 CT3EW2 59292007 IC50 > 1000 nM T64969 C2FYK8 59322489 IC50 = 82 nM T64969 C6NCJ4 59322491 IC50 = 7893 nM T64969 CS35WB 59322547 IC50 = 352 nM T64969 CN6PF7 59322583 IC50 = 589 nM T64969 CH5SO4 59322599 IC50 > 10000 nM T64969 C3KTW7 59322608 IC50 = 434 nM T64969 CGH6T7 59322651 IC50 = 179 nM T64969 CX2WH5 59322657 IC50 = 64 nM T64969 C9AEM1 59322682 IC50 = 218 nM T64969 C19QYP 59322697 IC50 = 3.9 nM T64969 C0YG3I 59322699 IC50 = 9 nM T64969 C9GWZ0 59322716 IC50 = 258 nM T64969 C52WSD 59322732 IC50 = 0.214 nM T64969 C67WFH 59322756 IC50 = 159 nM T64969 C7PE3G 59453176 IC50 = 6.9 nM T64969 CHC3W6 59484610 IC50 = 38 nM T64969 C1B3NR 59484612 IC50 = 110 nM T64969 CX0KC2 59484694 IC50 = 75 nM T64969 CXJ63M 59603829 IC50 = 28000 nM T64969 CQEU96 59603842 IC50 = 340 nM T64969 CXG78H 60020799 IC50 = 2991 nM T64969 C1MR8Q 60097495 IC50 > 1000 nM T64969 CSZA16 60155724 IC50 = 410 nM T64969 CK8EN9 60166357 IC50 = 59 nM T64969 CU79HD 60202383 IC50 = 2 nM T64969 C9ZCT2 62705065 IC50 > 1000 nM T64969 CUBL90 66545750 IC50 = 1620 nM T64969 CY5KC6 66550688 IC50 = 230 nM T64969 C4K2VC 66550892 IC50 = 1350 nM T64969 CK6WO0 66552478 IC50 < 10000 nM T64969 C10AMI 66553589 IC50 > 10000 nM T64969 C7CW0V 66554568 IC50 = 104.7 nM T64969 CPT48Z 66554916 IC50 = 167.3 nM T64969 C9ABY5 66555108 IC50 = 32.2 nM T64969 CID49H 66555110 IC50 = 5.8 nM T64969 C1FZ9G 66555254 IC50 = 100.1 nM T64969 CA2MK9 66555427 IC50 = 72.2 nM T64969 CB5RC1 66555609 IC50 > 1000 nM T64969 CE0U3J 66555781 IC50 = 1.8 nM T64969 CY6LN5 66555942 IC50 > 1000 nM T64969 C8N5KT 66555946 IC50 = 195.8 nM T64969 CQ61CB 66556107 IC50 = 102.2 nM T64969 CH35UQ 66556108 IC50 = 115.1 nM T64969 CXI2E5 66556610 IC50 = 121.1 nM T64969 CF5A3X 66556780 IC50 = 8.1 nM T64969 CRDU73 66556783 IC50 = 134.9 nM T64969 CWSJ26 66556966 IC50 = 560.4 nM T64969 C9QF6B 66559005 IC50 = 27 nM T64969 C1HSE0 67035086 IC50 = 2300 nM T64969 CWI6K5 67035106 IC50 > 10000 nM T64969 C38RGB 67035556 IC50 > 10000 nM T64969 CV3HW2 67035568 IC50 > 10000 nM T64969 CD14OC 67071561 IC50 = 3081 nM T64969 CEKN37 67073846 IC50 = 178 nM T64969 CR8L3N 67128637 IC50 = 3150 nM T64969 C7B9GO 67128667 IC50 = 8870 nM T64969 CWT14V 67137892 IC50 = 63.4 nM T64969 CV63UL 67240318 IC50 > 10000 nM T64969 C5SYC3 67304928 IC50 = 170 nM T64969 CR1ZL0 67346310 IC50 = 25 nM T64969 CCAD76 68196023 IC50 = 41 nM T64969 C8I7GC 68293638 IC50 > 10000 nM T64969 CD56XK 68293660 IC50 > 10000 nM T64969 CU57RD 68304261 IC50 > 25000 nM T64969 CI0A4N 68304989 IC50 = 400 nM T64969 C76TLN 68305106 IC50 = 630 nM T64969 C1FD5A 68342470 IC50 = 3100 nM T64969 C7WP9L 68342530 IC50 = 1700 nM T64969 C3JE5H 68356029 IC50 = 285 nM T64969 CNC27X 68594933 IC50 = 203 nM T64969 C57ENP 68629464 IC50 = 3 nM T64969 CG7KR4 68669354 IC50 = 9.8 nM T64969 CZB4E9 68672618 Ki = 22 nM T64969 CBIL54 68678227 IC50 > 10000 nM T64969 CAIO65 68796885 IC50 = 112 nM T64969 C5DGR9 69036886 IC50 = 10000 nM T64969 CW0E7O 69104616 IC50 = 257 nM T64969 CVN97F 69714349 IC50 = 109 nM T64969 CE5U7A 69956412 IC50 = 130016.96 nM T64969 C73ZTD 70023804 IC50 > 100000 nM T64969 C7IZW8 70681324 IC50 = 11 nM T64969 CK2G8E 70681325 IC50 = 0.49 nM T64969 CXRF43 70681934 IC50 = 2340 nM T64969 CLK09M 70681935 IC50 = 1800 nM T64969 CX5VN1 70681936 IC50 = 6170 nM T64969 C1ALW8 70682361 IC50 = 30000 nM T64969 CXW0E5 70682363 IC50 = 4500 nM T64969 CT5R9G 70682364 IC50 = 65000 nM T64969 CGM71F 70683719 IC50 = 0.29 nM T64969 CE3VQ2 70683720 IC50 = 0.68 nM T64969 C6USH3 70683721 IC50 = 37.5 nM T64969 CS30XY 70684051 IC50 = 1410 nM T64969 C9OT4C 70684052 IC50 = 1410 nM T64969 C5FYX7 70684449 IC50 = 1400 nM T64969 CJ83GE 70684450 IC50 = 6800 nM T64969 CNI19U 70684611 IC50 = 790 nM T64969 CDT70C 70684612 IC50 = 1290 nM T64969 C5DN2W 70684613 IC50 = 630 nM T64969 C9J0BO 70684614 IC50 = 216 nM T64969 CK83NM 70685870 IC50 = 17.4 nM T64969 C0JV2Y 70685871 IC50 = 2.21 nM T64969 C4M2OY 70686190 IC50 = 2220 nM T64969 CQE6H8 70686191 IC50 = 3530 nM T64969 CLT47X 70686585 IC50 = 230 nM T64969 CEV43U 70686586 IC50 = 140 nM T64969 CR5NW7 70686587 IC50 = 3000 nM T64969 C7L5MA 70686588 IC50 = 7800 nM T64969 CVH29P 70686589 IC50 = 120 nM T64969 C82FIP 70686752 IC50 = 700 nM T64969 CVP42W 70686767 IC50 = 1630 nM T64969 C7EM5X 70686945 IC50 = 120 nM T64969 CKCU42 70687611 IC50 > 10000 nM T64969 CE8LV1 70688705 IC50 = 61 nM T64969 C0QX3Y 70688829 IC50 = 510 nM T64969 CYP97H 70688851 IC50 = 570 nM T64969 C47IRO 70688852 IC50 = 1140 nM T64969 CDI67X 70689230 IC50 = 419 nM T64969 C24TEK 70690021 IC50 = 0.27 nM T64969 CC3D2S 70690022 IC50 = 1.46 nM T64969 C8KS2X 70690332 IC50 = 4200 nM T64969 C29RZD 70690333 IC50 = 2250 nM T64969 CM9C6X 70690334 IC50 = 900 nM T64969 C57QVT 70690769 IC50 = 78 nM T64969 C1OLS7 70690770 IC50 = 5800 nM T64969 CCT2Z7 70690771 IC50 = 75000 nM T64969 CT6CN0 70690772 IC50 = 570 nM T64969 CIJ57N 70690773 IC50 = 79000 nM T64969 CEQP73 70690935 IC50 = 98 nM T64969 CF30HQ 70692178 IC50 = 2.02 nM T64969 CXG2I4 70692907 IC50 = 380 nM T64969 CBS26Q 70692909 IC50 = 67 nM T64969 CH85TX 70692910 IC50 = 7200 nM T64969 CSOT12 70693058 IC50 > 10000 nM T64969 CS6NW3 70693059 IC50 > 10000 nM T64969 CR67GN 70693078 IC50 = 3680 nM T64969 CUT1L7 70693079 IC50 = 920 nM T64969 C1SF0B 70693242 IC50 = 5 nM T64969 CQ5W6D 70693519 IC50 = 6 nM T64969 C4N6ZM 70693874 IC50 > 10000 nM T64969 CS64HU 70694243 IC50 = 0.18 nM T64969 C68TLE 70694244 IC50 = 0.51 nM T64969 CP4V0G 70694245 IC50 = 50.7 nM T64969 CO1MU8 70694542 IC50 = 1100 nM T64969 C9D4UF 70694543 IC50 = 1120 nM T64969 CA0CP1 70694544 IC50 = 5160 nM T64969 CWM62Q 70694846 Ki > 10000 nM T64969 CHF7G6 70694948 IC50 = 3700 nM T64969 CI52UN 70695327 IC50 = 7 nM T64969 C6HI8Q 70696598 IC50 = 3310 nM T64969 CBCF23 70696599 IC50 = 1560 nM T64969 CW8A5I 70697001 IC50 = 380 nM T64969 C59NUJ 70697002 IC50 = 990 nM T64969 CWDR98 70697003 IC50 = 99 nM T64969 C3JW4Q 70697004 IC50 = 1700 nM T64969 C65CEI 70697160 IC50 = 2750 nM T64969 CH0B8N 70789756 IC50 > 30000 nM T64969 C5ILD4 70856339 IC50 = 91 nM T64969 CAI74T 70856585 IC50 = 10 nM T64969 C6W1NL 71244639 IC50 = 0.26 nM T64969 C5RE4T 71244643 IC50 = 0.27 nM T64969 CQ6A9L 71244644 IC50 = 0.53 nM T64969 CHT4N1 71244646 IC50 = 0.67 nM T64969 CH29GF 71258526 IC50 > 50000 nM T64969 C3BSP5 71449334 IC50 > 8000 nM T64969 C1LH2U 71449341 IC50 = 31 nM T64969 C4BXY8 71449342 IC50 = 56 nM T64969 C58BSC 71451912 IC50 = 631 nM T64969 CEBO91 71452977 IC50 = 11 nM T64969 C3MYB5 71453818 IC50 = 60 nM T64969 CJ2L8G 71455836 IC50 > 40000 nM T64969 CKT60L 71455860 Ki > 1800 nM T64969 CCGJ48 71456241 IC50 = 719 nM T64969 C7X4MD 71456750 IC50 = 10490 nM T64969 C9TZK4 71457259 IC50 = 215 nM T64969 CTWX94 71457629 IC50 > 40000 nM T64969 C3AEL4 71457630 IC50 > 40000 nM T64969 C4V6TN 71459522 IC50 > 40000 nM T64969 CEM84S 71462713 IC50 = 30 nM T64969 C7LCS8 71470563 IC50 = 12 nM T64969 CO0U6L 71473856 IC50 = 1 nM T64969 CMEH30 71473900 IC50 = 140 nM T64969 CH8NC9 71473954 IC50 = 78 nM T64969 C2PMJ7 71474167 IC50 = 4 nM T64969 CCR8J9 71496459 IC50 = 45 nM T64969 C8V4GQ 71496460 IC50 = 2 nM T64969 CQY31T 71498139 IC50 > 10000 nM T64969 C5AP8X 71508607 IC50 = 1600 nM T64969 CXQ43R 71508608 IC50 = 2200 nM T64969 CK13HD 71508609 IC50 = 1500 nM T64969 CJM0L4 71508610 IC50 = 2100 nM T64969 C2QTI4 71508643 IC50 = 8000 nM T64969 C3E4LW 71508644 IC50 = 6800 nM T64969 CQ2BV1 71508645 IC50 = 7100 nM T64969 COB85T 71508646 IC50 = 5600 nM T64969 CV6PN7 71508647 IC50 = 15300 nM T64969 CN5KQ8 71508648 IC50 = 7500 nM T64969 CDJB35 71508649 IC50 = 6100 nM T64969 CY60ZX 71508689 IC50 = 400 nM T64969 C21ZUC 71508690 IC50 = 20800 nM T64969 CSM31W 71508691 IC50 = 4600 nM T64969 C7FXT5 71508692 IC50 = 3900 nM T64969 CHZM56 71508693 IC50 = 5300 nM T64969 CK52TP 71508694 IC50 = 18600 nM T64969 C9TRM0 71508695 IC50 = 2000 nM T64969 CUHL20 71508717 IC50 = 1900 nM T64969 CY8QX5 71508718 IC50 = 4800 nM T64969 C9DIK2 71512060 IC50 = 0.2 nM T64969 C2VI1N 71512261 IC50 = 2.6 nM T64969 CF05BU 71513157 IC50 = 0.16 nM T64969 CS1ZX0 71513822 IC50 = 0.18 nM T64969 C2GP7V 71513823 IC50 = 0.89 nM T64969 CWX8Y4 71514053 IC50 = 0.3 nM T64969 CW6DN0 71514054 IC50 = 0.31 nM T64969 CXRK32 71519007 IC50 > 200 ug.mL-1 T64969 CI2Z5Y 71519008 IC50 > 200 ug.mL-1 T64969 CJ4KV6 71519009 IC50 > 200 ug.mL-1 T64969 C42MFK 71519172 IC50 > 200 ug.mL-1 T64969 C3XP1F 71519173 IC50 = 94 ug.mL-1 T64969 CC89QU 71519174 IC50 = 120 ug.mL-1 T64969 CGY2N8 71519175 IC50 > 200 ug.mL-1 T64969 C7RG1Z 71519338 IC50 = 193 ug.mL-1 T64969 COFB13 71519339 IC50 = 130 ug.mL-1 T64969 CJE5N6 71519340 IC50 = 130 ug.mL-1 T64969 CG0N8I 71519341 IC50 = 148 ug.mL-1 T64969 CM4PG6 71519493 IC50 > 200 ug.mL-1 T64969 CVUP53 71524867 IC50 = 2230 nM T64969 CQ52FW 71524868 IC50 = 8250 nM T64969 CQ7L5U 71524869 IC50 = 940 nM T64969 CVPO31 71524870 IC50 = 5680 nM T64969 CSM8Q3 71524871 IC50 = 160 nM T64969 CHZA07 71524872 IC50 = 2060 nM T64969 CW9M5E 71524873 IC50 = 210 nM T64969 C75GEB 71524914 IC50 = 3010 nM T64969 CO1H9P 71524915 IC50 = 3280 nM T64969 CNZF95 71524916 IC50 = 1070 nM T64969 CXP7G2 71524917 IC50 = 680 nM T64969 CQR8V0 71524918 IC50 = 490 nM T64969 CQ34CK 71524919 IC50 = 100 nM T64969 C12GMV 71524960 IC50 = 140 nM T64969 C7BU0K 71524961 IC50 = 300 nM T64969 C4R6CL 71524962 IC50 = 530 nM T64969 CQ7UT5 71524963 IC50 = 350 nM T64969 CRO0N8 71524964 IC50 = 1040 nM T64969 CZQ2S4 71524965 IC50 = 520 nM T64969 C8A9IN 71525006 IC50 = 660 nM T64969 CH8LC0 71525007 IC50 = 710 nM T64969 CT47DK 71525008 IC50 = 120 nM T64969 C0M4LC 71525009 IC50 = 50 nM T64969 C5OBF0 71525245 IC50 = 85900 nM T64969 CJX73B 71525246 IC50 = 110600 nM T64969 CCN90I 71525247 IC50 = 19900 nM T64969 CY6JA9 71525248 IC50 = 19300 nM T64969 CGQJ60 71525249 IC50 = 15600 nM T64969 CMKD15 71525283 IC50 = 5400 nM T64969 C3OJ6R 71525284 IC50 = 16300 nM T64969 CP5Q2U 71525285 IC50 > 200000 nM T64969 CZ8N0J 71525286 IC50 = 12800 nM T64969 CG31MI 71525287 IC50 = 26900 nM T64969 C1SFD7 71532857 IC50 > 200 ug.mL-1 T64969 C8U9MB 71532907 IC50 > 200 ug.mL-1 T64969 COQ5V1 71532908 IC50 > 200 ug.mL-1 T64969 CE9N2D 71532909 IC50 > 200 ug.mL-1 T64969 C1D3KG 71535003 Ki = 4 nM T64969 CS2X3D 71535296 Ki = 3 nM T64969 CN4AW3 71543353 IC50 = 6.1 nM T64969 CCN01X 71547862 IC50 > 10000 nM T64969 C2NLX4 71549099 IC50 = 2.7 nM T64969 CA3O6K 71552696 IC50 > 30000 nM T64969 C1NPL0 71552941 IC50 = 4290 nM T64969 CA4PS8 71552942 IC50 = 4090 nM T64969 C3UA9C 71553011 IC50 = 30000 nM T64969 CEZ15Y 71553012 IC50 = 30000 nM T64969 CVIA91 71553085 IC50 = 30000 nM T64969 C1TR3O 71553152 IC50 = 30000 nM T64969 CVNA30 71558752 IC50 > 5000 nM T64969 CEJ97M 71558906 IC50 = 600 nM T64969 C1L8GW 71558907 IC50 = 600 nM T64969 CI6QF8 71571535 IC50 = 8 nM T64969 CT4O9F 71571536 IC50 = 29 nM T64969 CRX81Q 71575642 IC50 > 10000 nM T64969 CN9BQ0 71579162 IC50 = 61 nM T64969 CN7W5S 71579325 IC50 = 126.7 nM T64969 CA9KL5 71579403 IC50 = 12.1 nM T64969 CMV9U3 71579405 IC50 = 13.6 nM T64969 C1BCX0 71579696 IC50 > 1000 nM T64969 CGK76E 71583411 IC50 > 200000 nM T64969 CB5WX0 71583412 IC50 = 42000 nM T64969 CI8K3T 71583527 IC50 = 63600 nM T64969 C6FGI0 71583528 IC50 = 38900 nM T64969 C3QGE7 71583529 IC50 > 200000 nM T64969 CS9HX7 71583530 IC50 = 114700 nM T64969 CQTZ32 71583531 IC50 = 39200 nM T64969 C0G5RS 71583532 IC50 = 58700 nM T64969 CVEY46 71583533 IC50 > 200000 nM T64969 CX6TR7 71583634 IC50 = 30800 nM T64969 CR15QP 71583635 IC50 = 130500 nM T64969 CZ31PU 71583657 IC50 = 36 nM T64969 C6RS7H 71583658 IC50 = 47 nM T64969 CWD2Z5 71585566 IC50 = 4 nM T64969 CCE7T2 71585568 IC50 = 3610 nM T64969 CO32SN 71599995 IC50 = 15 nM T64969 CQS51R 71615916 IC50 = 16 nM T64969 C4KUE9 71616518 IC50 = 56 nM T64969 CQX8L3 71616700 IC50 = 4.3 nM T64969 CE6QA1 71616701 IC50 = 3 nM T64969 C4ZDO0 71616702 IC50 = 7.4 nM T64969 C03HCR 71616703 IC50 = 0.3 nM T64969 CWTH52 71616704 IC50 = 0.5 nM T64969 CZ7XB4 71616807 IC50 = 22 nM T64969 C9YLM0 71621675 IC50 = 30 nM T64969 CH2RA9 71658877 IC50 > 5000 nM T64969 CJI05L 71658878 IC50 = 460 nM T64969 CCS41V 71658995 IC50 = 45 nM T64969 CK10SJ 71658996 IC50 > 5000 nM T64969 CI91ZX 71658997 IC50 > 5000 nM T64969 CL9T2I 71658998 IC50 > 5000 nM T64969 C1JZG9 71658999 IC50 = 1500 nM T64969 CKMO02 71659116 IC50 > 5000 nM T64969 CY5VP3 71659117 IC50 > 5000 nM T64969 CG21JR 71659118 IC50 = 2300 nM T64969 C0LHW7 71659119 IC50 = 660 nM T64969 C2IS8V 71659241 IC50 = 2500 nM T64969 C78PSE 71659242 IC50 = 3500 nM T64969 CB4LV9 71659243 IC50 = 3000 nM T64969 CGB5L8 71659244 IC50 > 5000 nM T64969 C45CVT 71659245 IC50 > 5000 nM T64969 CC6L2A 71659371 IC50 = 850 nM T64969 CQV2I4 71659372 IC50 = 900 nM T64969 CC9F0T 71659373 IC50 = 2000 nM T64969 CEBL45 71659374 IC50 = 5500 nM T64969 CHM79O 71659375 IC50 = 6000 nM T64969 CX46VT 71659505 IC50 = 5000 nM T64969 C0Y3VS 71659506 IC50 = 800 nM T64969 C3A8IH 71659507 IC50 = 1000 nM T64969 C2MS9Y 71659508 IC50 = 1500 nM T64969 C64SFQ 71659509 IC50 = 5000 nM T64969 CN6LI7 71659629 IC50 = 4500 nM T64969 C7TAL4 71659630 IC50 = 800 nM T64969 C82HXJ 71659631 IC50 = 1200 nM T64969 C2A8VJ 71659632 IC50 = 3500 nM T64969 CU27RN 71659633 IC50 = 6000 nM T64969 C2ZRK6 71659769 IC50 = 450 nM T64969 C8XM3E 71659770 IC50 = 600 nM T64969 CT79UA 71659771 IC50 = 5000 nM T64969 C6AP4D 71659772 IC50 = 6000 nM T64969 CWQ09K 71661337 IC50 = 48 nM T64969 CIK32R 71661338 IC50 = 34 nM T64969 C9PGV4 71661339 IC50 = 4327 nM T64969 CKZ6B3 71661527 IC50 > 25000 nM T64969 C1FAU8 71679855 IC50 > 100000 nM T64969 CGU2J5 71680740 IC50 = 13 nM T64969 CEWI73 71680741 IC50 = 6 nM T64969 C6K5HT 71680742 IC50 = 42 nM T64969 CFLZ59 71680901 IC50 = 20 nM T64969 CU3E6I 71680902 IC50 = 17 nM T64969 C80AGF 71680903 IC50 = 23 nM T64969 CNC9S6 71681062 IC50 = 38 nM T64969 C9TZN5 71681063 IC50 = 16 nM T64969 CT4A0M 71681064 IC50 = 101 nM T64969 CRZ1F9 71681212 IC50 = 47 nM T64969 CZ1IO5 71683105 IC50 = 14 nM T64969 CST14N 71717689 IC50 = 147 nM T64969 C1JBD5 71720447 IC50 = 4.6 nM T64969 CED2H8 71720674 IC50 = 4700 nM T64969 C30NBJ 71722055 IC50 = 2100 nM T64969 C9Z0KG 71726907 IC50 = 13 nM T64969 C4X1CP 71748056 IC50 = 874 nM T64969 C07EWM 71761646 IC50 = 17.2 nM T64969 CMO51F 71761647 IC50 = 76 nM T64969 CR08OT 71762114 IC50 = 8.4 nM T64969 CSWH95 72164480 IC50 = 4100 nM T64969 CFUD13 72164482 IC50 = 3400 nM T64969 C7P0NM 72164483 IC50 = 1500 nM T64969 C0M8QJ 72164486 IC50 = 5100 nM T64969 CD7G1S 72164602 IC50 = 4700 nM T64969 CTC7H5 72164605 IC50 = 2400 nM T64969 C5X1DO 72164726 IC50 = 3600 nM T64969 CSA2J6 72187684 IC50 = 0.677 nM T64969 CX0N2A 72189794 IC50 = 0.63 nM T64969 CZ3XL6 72190112 IC50 = 0.41 nM T64969 CSK78J 72190113 IC50 = 19 nM T64969 CF4TJ9 72191350 IC50 = 190 nM T64969 CP2OR8 72191351 IC50 = 52 nM T64969 CM1B2Y 72191352 IC50 = 158 nM T64969 C5L0BJ 72191353 IC50 = 26 nM T64969 C4J3KE 72191667 IC50 = 94 nM T64969 C4DQ3P 72191668 IC50 = 36 nM T64969 C1YC7S 72191669 IC50 = 48 nM T64969 CNMJ61 72191670 IC50 = 24 nM T64969 C2MQ6X 72191671 IC50 = 25 nM T64969 CEB67M 72191672 IC50 = 34 nM T64969 C7V8MX 72195043 IC50 = 6 nM T64969 C1R7VY 72195184 IC50 = 8.1 nM T64969 CQR2N5 72201345 IC50 = 1.2 nM T64969 CC2X5T 72201349 IC50 = 0.5 nM T64969 CF75TB 72201501 IC50 = 4 nM T64969 CFA2J9 72201502 IC50 = 6.7 nM T64969 CIU90H 72202607 IC50 = 16 nM T64969 C4N9OI 72202732 IC50 = 1.07 nM T64969 CKAF40 72202733 IC50 = 33885 nM T64969 C7FJB9 72202734 IC50 = 13.8 nM T64969 CSW20D 72202735 IC50 = 4.53 nM T64969 CYB05D 72202865 IC50 = 3.97 nM T64969 C2MY1Q 72202866 IC50 = 6754 nM T64969 CV23JN 72202867 IC50 = 4.96 nM T64969 CW8HV3 72202868 IC50 = 4.72 nM T64969 C6FZA2 72202870 IC50 = 17.6 nM T64969 COK12B 72202930 IC50 = 0.5 nM T64969 CI3B4N 72202931 IC50 = 0.2 nM T64969 C8WC6P 72202999 IC50 = 4.94 nM T64969 C1TIX3 72203001 IC50 = 60.4 nM T64969 CW18BO 72203003 IC50 = 6.95 nM T64969 CI63WE 72203004 IC50 = 691 nM T64969 CYT82Q 72203134 IC50 = 39.7 nM T64969 C0K6SQ 72203136 IC50 = 26283 nM T64969 C7MV3O 72203732 IC50 = 250 nM T64969 CYB30W 72203733 IC50 = 410 nM T64969 C90ZBE 72203734 IC50 = 19 nM T64969 C5EWB0 72203735 IC50 = 68 nM T64969 C6KB7T 72203914 IC50 = 45 nM T64969 C9Q6LM 72206524 IC50 = 780 nM T64969 CKH1F8 72206525 IC50 = 960 nM T64969 CUT5W6 72206526 IC50 = 140 nM T64969 CE1VK7 72543781 IC50 = 13200 nM T64969 CLM4G2 72543782 IC50 = 9800 nM T64969 CF9LG1 72543783 IC50 = 31400 nM T64969 C3AT2E 72543784 IC50 = 3100 nM T64969 C32RMJ 72544014 IC50 = 7400 nM T64969 C7J4XV 72544015 IC50 = 6500 nM T64969 CPL35N 72544251 IC50 = 7600 nM T64969 CNT79J 72545791 IC50 = 10020 nM T64969 CN89UW 72545792 IC50 = 6130 nM T64969 CGY75C 72545793 IC50 = 12450 nM T64969 C8U6KH 72546029 IC50 = 2580 nM T64969 CW4VL8 72546030 IC50 = 1890 nM T64969 COR35N 72546031 IC50 = 210 nM T64969 CC9VQ1 72546032 IC50 = 430 nM T64969 C5QZS6 72546033 IC50 = 8190 nM T64969 CAM91I 72547360 IC50 = 8100 nM T64969 CEZQ57 72697432 IC50 = 1230 nM T64969 CL7A4Z 72697433 IC50 = 1180 nM T64969 CUD9M1 72697435 IC50 = 3510 nM T64969 C4AWS3 72697576 IC50 = 5490 nM T64969 C5M3GE 72697580 IC50 = 2120 nM T64969 COX45Z 72697720 IC50 = 3060 nM T64969 C10VYB 72697722 IC50 = 1380 nM T64969 CJ7E1C 72699656 IC50 = 4 nM T64969 CF4D5O 72699657 IC50 = 10 nM T64969 C52NAB 72699658 IC50 > 50000 nM T64969 C64UEN 72699659 IC50 > 32770 nM T64969 CKPL31 72700004 IC50 = 6810 nM T64969 C90VOI 72700006 IC50 = 50 nM T64969 CA4M7U 72700007 IC50 > 50000 nM T64969 CWZG30 72700008 IC50 > 50000 nM T64969 CG7AI6 72700079 IC50 > 50000 nM T64969 CI8ZY3 72700080 IC50 > 50000 nM T64969 CWRL78 72700165 IC50 = 4 nM T64969 CWBC84 72703789 IC50 = 421 nM T64969 CM75FY 72703989 IC50 = 68 nM T64969 CPQ34Z 72703991 IC50 = 72 nM T64969 CYG95S 72707651 IC50 > 5000 nM T64969 CNP0V5 72707724 IC50 > 5000 nM T64969 CU4A5Q 72707728 IC50 > 5000 nM T64969 CZAM98 72707790 IC50 > 5000 nM T64969 CP13FK 72707853 IC50 > 5000 nM T64969 C9OQ2I 72710839 IC50 > 10000 nM T64969 C26NTQ 72712708 IC50 = 708.5 nM T64969 CBN20W 72712709 IC50 = 143.6 nM T64969 C1XO0R 72712710 IC50 > 1000 nM T64969 CQ96FB 72712711 IC50 = 525 nM T64969 CEF73D 72712712 IC50 = 864 nM T64969 C4BX2Y 72712713 IC50 = 58.7 nM T64969 C01QBS 72712714 IC50 = 42.9 nM T64969 CAZ9P0 72712883 IC50 = 40.3 nM T64969 CA26ZY 72712884 IC50 = 204.1 nM T64969 CVH9B7 72712885 IC50 = 107.1 nM T64969 C9R5TW 72712886 IC50 = 8.8 nM T64969 CWI13Y 72712887 IC50 = 15.2 nM T64969 C9F8WM 72712888 IC50 = 235.4 nM T64969 CO7YX5 72712889 IC50 = 29.1 nM T64969 C2GRZ1 72712890 IC50 = 97.9 nM T64969 CX9L1B 72712891 IC50 = 16.2 nM T64969 C8R5SM 72712892 IC50 = 41.3 nM T64969 CRI42Q 72712893 IC50 = 7.2 nM T64969 CLX3M1 72712894 IC50 = 17.1 nM T64969 CSNU50 72712895 IC50 = 55.5 nM T64969 C54LQO 72712896 IC50 = 35.6 nM T64969 CY56SR 72712897 IC50 = 9.2 nM T64969 CUS2R1 72712978 IC50 = 21280 nM T64969 C87MUD 72712979 IC50 = 3836 nM T64969 C5ZU4Y 72713172 IC50 = 4802 nM T64969 CUDS15 72713174 IC50 = 31.3 nM T64969 CH93FM 72713175 IC50 = 373.5 nM T64969 CH3K0R 72713176 IC50 = 5585 nM T64969 C9LA5P 72713177 IC50 = 5.12 nM T64969 CK3N8G 72713385 IC50 = 272 nM T64969 CXU6R4 72713386 IC50 = 16338 nM T64969 CGN60W 72713387 IC50 = 5.29 nM T64969 CPA37Q 72734868 IC50 = 464 nM T64969 CJE91U 72734869 IC50 = 699 nM T64969 C2ZP3W 72734870 IC50 = 859 nM T64969 CWQ1G5 72734871 IC50 = 884 nM T64969 C0AVR4 72734872 IC50 = 1715 nM T64969 CSDQ79 72735047 IC50 = 265 nM T64969 CW3HI2 72735048 IC50 = 304 nM T64969 CG82VX 72735049 IC50 = 331 nM T64969 CKU16J 72735050 IC50 = 232 nM T64969 CFM8W4 72735051 IC50 = 404 nM T64969 CI2YH8 72737033 IC50 = 27 nM T64969 CE7T5Y 72737034 IC50 = 479 nM T64969 CIDN27 72737035 IC50 = 41 nM T64969 CTC3I9 72737206 IC50 = 635 nM T64969 C6QFZ8 72737207 IC50 = 365 nM T64969 C60TUV 72737208 IC50 = 68 nM T64969 CZ7U9H 72737209 IC50 = 165 nM T64969 CNX58O 72737210 IC50 = 82 nM T64969 CZ4IY1 72737401 IC50 = 197 nM T64969 CC38YI 72737402 IC50 = 544 nM T64969 C4SRQ7 72737403 IC50 = 24 nM T64969 CJ3WA6 72737404 IC50 = 32 nM T64969 CL7WI5 72737405 IC50 = 281 nM T64969 C8ADG7 72737575 IC50 = 505 nM T64969 CU9PS0 72737576 IC50 = 464 nM T64969 C8IV1S 72737577 IC50 = 543 nM T64969 C2S1ZE 72737578 IC50 = 967 nM T64969 C20NFB 72737579 IC50 = 1581 nM T64969 CQF4K5 72950786 IC50 = 0.79 nM T64969 CP58UB 73053605 IC50 = 3 nM T64969 C89HEJ 73291830 IC50 = 250 nM T64969 C5LGB4 73291831 IC50 = 220 nM T64969 CWC12F 73291832 IC50 = 290 nM T64969 C4B1CL 73291833 IC50 = 15200 nM T64969 CG8RI0 73292361 IC50 = 19 nM T64969 CC16IJ 73292362 IC50 = 19000 nM T64969 C7LPO0 73292363 IC50 = 5.6 nM T64969 CBQ72N 73292545 IC50 = 63 nM T64969 C9M7EL 73294313 IC50 = 770 nM T64969 CED6P2 73294314 IC50 = 81 nM T64969 CTPF92 73294315 IC50 = 22 nM T64969 C87AQU 73294502 IC50 = 12900 nM T64969 CDM86C 73294503 IC50 = 2100 nM T64969 C0D5EA 73294504 IC50 = 2800 nM T64969 C2UB8T 73294505 IC50 = 33 nM T64969 CAU94B 73294506 IC50 = 1550 nM T64969 CQV1P0 73294507 IC50 = 91 nM T64969 C3MF2U 73335400 IC50 = 9 nM T64969 C3QEG6 73335403 IC50 = 72 nM T64969 CE25BK 73335501 IC50 = 27 nM T64969 CZ90QC 73335502 IC50 = 32 nM T64969 CZP84O 73335598 IC50 > 10000 nM T64969 CJ3BK2 73335600 IC50 = 34 nM T64969 C06IFC 73335691 IC50 = 390 nM T64969 CC4DW1 73335692 IC50 = 33 nM T64969 C9JS7Z 73335693 IC50 = 880 nM T64969 C43EUZ 73335785 IC50 = 27 nM T64969 C0HSC8 73346520 Ki = 6090 nM T64969 C8SD9P 73346521 Ki = 55290 nM T64969 CGZ6Y8 73346522 Ki = 6640 nM T64969 C18WCY 73346557 IC50 = 1.29 nM T64969 C41QZC 73347162 Ki = 4000 nM T64969 C43IPQ 73348006 Ki = 15650 nM T64969 C8SIL6 73349435 IC50 = 90.05 nM T64969 CV21FR 73349643 IC50 = 100 nM T64969 C9EXR4 73351100 IC50 = 21.1 nM T64969 CS9C0W 73351108 Ki = 27400 nM T64969 CXC0O2 73352566 IC50 = 25.1 nM T64969 CZJ2S7 73352567 IC50 = 18.7 nM T64969 CCI47S 73352568 IC50 = 10.8 nM T64969 C27JUH 73352576 Ki = 8580 nM T64969 CVP03Z 73352577 Ki = 41580 nM T64969 CX75YR 73352604 IC50 = 630.96 nM T64969 C9TMA1 73352657 IC50 = 100 nM T64969 CDAB86 73354065 Ki = 2970 nM T64969 CK3Z8U 73354066 Ki = 4680 nM T64969 C92DXZ 73354067 Ki = 22940 nM T64969 C83XBD 73354112 IC50 = 7 nM T64969 CCI18Y 73355591 Ki = 5820 nM T64969 CRX8A0 73355592 Ki = 16770 nM T64969 C8XHK6 73356867 IC50 = 2300 nM T64969 CYQ8K1 73357210 IC50 = 70 nM T64969 CVNW01 73386831 IC50 > 1000 nM T64969 CQ5E3H 73707531 IC50 = 16.8 nM T64969 CX1LR9 73774633 IC50 = 26 nM T64969 CS9BQ1 74222426 IC50 = 3890 nM T64969 CO0V6K 74222427 IC50 = 16800 nM T64969 CBE71O 74222509 IC50 > 20000 nM T64969 CM02PA 74222510 IC50 = 1710 nM T64969 CWLT81 74222511 IC50 > 20000 nM T64969 C4XSG8 74222512 IC50 = 274 nM T64969 CBT4M6 74222513 IC50 = 2180 nM T64969 C53AFH 74222599 IC50 = 2910 nM T64969 CNR7C1 74223711 IC50 = 126.3 nM T64969 CJ0N5V 74223816 IC50 = 1.06 nM T64969 CF9A7B 74766095 Ki = 2 nM T64969 CM1VR8 74766099 Ki = 0.14 nM T64969 C4WHJ6 74937126 IC50 = 1 nM T64969 C97KTL 76007179 IC50 = 34.16 nM T64969 C7K2QN 76280903 Ki = 22 nM T64969 CP1W6F 76281713 Ki = 151 nM T64969 CN1RJ8 76282701 Ki = 18 nM T64969 C1XZY3 76282702 Ki = 14 nM T64969 CFP9O7 76309779 IC50 = 7300 nM T64969 CW5OG2 76310006 IC50 = 61500 nM T64969 C8DX4U 76311274 IC50 = 275 nM T64969 C0HX2E 76311275 IC50 = 53300 nM T64969 C07IBW 76312208 IC50 = 250034.54 nM T64969 CH24LB 76313481 IC50 = 130 nM T64969 C7MLX4 76313718 IC50 = 18300 nM T64969 CRV24X 76313719 IC50 > 100000 nM T64969 CW5A6P 76314206 IC50 > 10000 nM T64969 CDG1O5 76316997 IC50 = 200 nM T64969 C0M2LJ 76316998 IC50 = 1100 nM T64969 CZK2V6 76317238 IC50 > 100000 nM T64969 CKG8C3 76317239 IC50 = 34600 nM T64969 C27JRQ 76317764 IC50 = 4 nM T64969 C8AJ3M 76317765 IC50 = 3 nM T64969 C4PT8M 76318480 IC50 > 5000 nM T64969 CF06PR 76318481 IC50 = 2200 nM T64969 CK5UL0 76318482 IC50 = 2000 nM T64969 CE95GB 76318483 IC50 = 43700 nM T64969 CX7RD0 76320712 IC50 = 1200 nM T64969 CJE4B1 76321478 IC50 = 16 nM T64969 C13XBM 76321479 IC50 > 10000 nM T64969 CG29RA 76321480 IC50 > 10000 nM T64969 CLO8N7 76321481 IC50 > 10000 nM T64969 CG67DB 76321482 IC50 = 12 nM T64969 C6SCV7 76322145 IC50 = 3200 nM T64969 CL0T7B 76322219 IC50 = 2145 nM T64969 CPD3W5 76324607 IC50 = 1630 nM T64969 CZ6AK2 76325089 IC50 > 10000 nM T64969 CBP83A 76325766 IC50 = 2.1 nM T64969 C4K7IO 76325767 IC50 = 2300 nM T64969 C4RD8T 76325768 IC50 = 1.5 nM T64969 CH6V0B 76327248 IC50 = 12880 nM T64969 CHDR08 76327920 IC50 = 9 nM T64969 CPZN18 76328168 IC50 > 100000 nM T64969 CDP53X 76328653 IC50 > 10000 nM T64969 CE1L8A 76329348 IC50 = 931 nM T64969 CV4ZP1 76331568 IC50 = 33 nM T64969 CA45HZ 76331569 IC50 = 3 nM T64969 C0BJ8F 76332331 IC50 = 5 nM T64969 C83DTC 76332332 IC50 > 10000 nM T64969 CJ2T9E 76332983 IC50 = 270 nM T64969 CC25SV 76332992 IC50 = 9800 nM T64969 CS47NK 76332993 IC50 = 2800 nM T64969 C7K1PL 76332994 IC50 = 3950 nM T64969 COTE80 76332995 IC50 = 2500 nM T64969 C9GRT4 76332996 IC50 = 76500 nM T64969 CAP7F0 76335418 IC50 = 67200 nM T64969 C51LIY 76335419 IC50 > 100000 nM T64969 C4J5BS 76335961 IC50 = 5 nM T64969 C28UES 76335962 IC50 > 10000 nM T64969 CG56FE 76335963 IC50 = 82 nM T64969 CP3YE6 76336599 IC50 = 3710 nM T64969 C4V0GX 76336600 IC50 = 4400 nM T64969 CZR21Q 76336601 IC50 = 8730 nM T64969 C4QPA1 76336602 IC50 = 130 nM T64969 C2N9EB 76336603 IC50 = 2200 nM T64969 C4HOM3 76900440 IC50 = 1935 nM T64969 CT92YM 77461033 IC50 = 6 nM T64969 CH8W7D 77461036 IC50 > 1000 nM T64969 CWG4T2 78209992 IC50 < 0.5 nM T64969 CS8V1X 78318941 IC50 = 2.9 nM T64969 CA5SQ8 78319175 IC50 = 1 nM T64969 CH8XY3 78322920 IC50 > 10000 nM T64969 C2YSJ7 78323235 IC50 > 10000 nM T64969 CTJ02F 78323236 IC50 > 10000 nM T64969 C5P4JF 78323237 IC50 > 10000 nM T64969 CVZ26O 78323238 IC50 > 10000 nM T64969 CP90IE 78323239 IC50 = 890 nM T64969 CAZ2J6 78323563 IC50 = 1010 nM T64969 CXC01P 78323564 IC50 = 360 nM T64969 CGP5M8 78323565 IC50 > 10000 nM T64969 CNA52Z 78324176 IC50 = 9 nM T64969 C90PJT 78324177 IC50 = 3 nM T64969 CEDG87 78324478 IC50 = 5 nM T64969 C2JKT5 78324480 IC50 = 27 nM T64969 CQA2Y0 78324481 IC50 = 3 nM T64969 CT81NA 78324482 IC50 = 550 nM T64969 CV0P3A 78357783 IC50 = 200 nM T64969 C7CGZ1 85206710 IC50 = 800 nM T64969 CK61HY 85469442 IC50 > 10000 nM T64969 CL19KE 85471023 IC50 = 5.3 nM T64969 CYAS09 85471025 IC50 = 2.1 nM T64969 C93JAB 85471026 IC50 = 520.2 nM T64969 C97GER 85471045 IC50 = 356.6 nM T64969 C7YK6I 85471046 IC50 = 109.4 nM T64969 CD51LP 85471121 IC50 = 1.56 nM T64969 CRT9W7 85471122 IC50 = 1.3 nM T64969 CNXC02 85471147 IC50 = 4.5 nM T64969 CR1O7P 85471149 IC50 = 3.5 nM T64969 C2WLZ6 85827467 Ki = 700 nM T64969 CV4TL7 86276219 IC50 = 270 nM T64969 CH2X3O 86276220 IC50 = 21020 nM T64969 C8R4JZ 86276226 IC50 = 4100 nM T64969 CRA39W 86276227 IC50 = 180 nM T64969 C7QXC2 86276228 IC50 = 120 nM T64969 C7GE4I 86276229 IC50 = 420 nM T64969 CBQ9L7 86276271 IC50 < 0.25 nM T64969 CQ9H4U 86277844 IC50 = 7500 nM T64969 CV8UZ1 86278565 Ki = 17 nM T64969 CSH3G2 86287525 IC50 > 10000 nM T64969 C0QK9F 86288869 IC50 = 94 nM T64969 CWYE62 86294833 IC50 = 1320 nM T64969 CCJ43A 86302281 IC50 = 16 nM T64969 CH5AD6 86302282 IC50 = 9 nM T64969 CJL1W6 86302308 IC50 = 4 nM T64969 C7U3VF 86302309 IC50 = 3 nM T64969 CA72QE 86302441 IC50 = 510 nM T64969 CQ9J7S 86302442 IC50 = 10120 nM T64969 CB5NJ4 86302541 IC50 > 10000 nM T64969 CPG3A5 86302574 IC50 > 30000 nM T64969 C7MA0Y 86302767 IC50 = 444.7 nM T64969 C2L4GR 86303858 IC50 = 4 nM T64969 C08WGI 86566799 IC50 > 10000 nM T64969 C9NTP1 86677234 IC50 = 2000 nM T64969 CEKQ13 86677242 IC50 = 19000 nM T64969 C5YX8T 86677253 IC50 = 1000 nM T64969 CCX1U5 86677265 IC50 = 2000 nM T64969 CZQ1F7 86677270 IC50 = 311 nM T64969 CB5Z8H 86677276 IC50 < 1 nM T64969 C1KLC3 86679616 Ki = 3 nM T64969 CR08QT 89266687 IC50 = 550 nM T64969 CNZ86G 89456691 IC50 = 7.6 nM T64969 CP0MJ8 89456904 Ki = 35 nM T64969 CK78NF 89456980 Ki = 3 nM T64969 CY12PC 89457089 Ki = 8 nM T64969 CS42DR 89457109 Ki = 8 nM T64969 C32JOH 89457151 Ki = 4 nM T64969 C1HTP4 89457165 Ki = 4 nM T64969 CNSK27 89457251 Ki = 3 nM T64969 CR5QA1 89457296 IC50 = 1.6 nM T64969 CM8T1V 89556219 IC50 = 36 nM T64969 C1HW4B 89735655 IC50 > 100000 nM T64969 CR3XL7 90119070 IC50 > 20000 nM T64969 CLK3O0 90119255 IC50 = 570 nM T64969 CO2FV0 90119264 IC50 = 15 nM T64969 C3RL4C 90136268 IC50 > 20000 nM T64969 C4ME0V 90136282 IC50 = 15400 nM T64969 CY0T6O 90136348 IC50 = 149 nM T64969 CN2RJ1 90178371 Ki = 20 nM T64969 C5XEP6 90183257 Ki = 76 nM T64969 C70HZA 90183266 Ki = 201 nM T64969 C3G4AS 90183295 Ki = 149 nM T64969 CM6GB2 90183305 Ki = 19 nM T64969 C4DEJ1 90183313 Ki = 71 nM T64969 CHR3J1 90183333 Ki = 48 nM T64969 C70EWF 90183350 Ki = 87 nM T64969 CV64KY 90183363 Ki = 40 nM T64969 C1GZ4H 90183367 Ki = 19 nM T64969 CY3P2G 90183439 Ki = 124 nM T64969 CKQ87S 90183468 Ki = 27 nM T64969 C5HZ0I 90183471 Ki = 658 nM T64969 CIR8P9 90183483 Ki = 28 nM T64969 CD08SZ 90183490 Ki = 196 nM T64969 CL12RI 90183503 Ki = 323 nM T64969 C8NLP0 90183548 Ki = 329 nM T64969 C97YQB 90183560 Ki = 2.7 nM T64969 C7TQI0 90183635 Ki = 492 nM T64969 C7TKR1 90183640 Ki = 77 nM T64969 C03ZHC 90183641 Ki = 24 nM T64969 C9A4WX 90183658 Ki = 2.5 nM T64969 CR7CN0 90183696 Ki = 38 nM T64969 CON0U4 90183732 Ki = 50 nM T64969 CL4JO2 90183809 Ki = 33 nM T64969 C7DT2U 90183870 Ki > 0.53 nM T64969 C8BJ6V 90183913 Ki = 4.3 nM T64969 CX4L6E 90183992 Ki = 13 nM T64969 CWT70U 90185859 IC50 = 94 nM T64969 CZF18X 90185862 IC50 = 11 nM T64969 CAF0J8 90185892 IC50 = 1.3 nM T64969 C2QD8N 90185907 IC50 = 10 nM T64969 CIY1J5 90185909 IC50 = 19 nM T64969 CIT45C 90185926 IC50 = 39 nM T64969 CA6KX8 90185944 IC50 = 95 nM T64969 CK2NU8 90185982 IC50 = 78 nM T64969 C75IJT 90185983 IC50 = 23.5 nM T64969 CLT57U 90185984 IC50 = 20 nM T64969 CS6VQ3 90186050 IC50 = 17.8 nM T64969 CB9CG5 90282624 IC50 = 1 nM T64969 CPH85G 90322858 IC50 = 4 nM T64969 C1UQ3H 90375291 IC50 = 1.2 nM T64969 CF7XO6 90375389 IC50 = 63.8 nM T64969 C5S3YB 90645165 IC50 > 10000 nM T64969 CY0UC4 90645194 IC50 > 10000 nM T64969 C3GU7P 90645237 IC50 > 10000 nM T64969 CFI93O 90645239 IC50 > 10000 nM T64969 C76KSB 90645241 IC50 > 10000 nM T64969 CNWP80 90645243 IC50 > 10000 nM T64969 C1POJ2 90645244 IC50 > 10000 nM T64969 C8BEX4 90645245 IC50 > 10000 nM T64969 C6Q4DH 90645475 IC50 = 73.3 nM T64969 C89HTB 90645476 IC50 = 340.1 nM T64969 CL32MR 90645477 IC50 = 113.2 nM T64969 C9ASG1 90645478 IC50 = 70.7 nM T64969 COY53U 90645479 IC50 = 30 nM T64969 C48OSQ 90645480 IC50 = 84.4 nM T64969 CL8GW5 90645481 IC50 = 122.1 nM T64969 CL7SC6 90645482 IC50 = 90.2 nM T64969 C5U6RM 90645483 IC50 = 30.2 nM T64969 CI3OD6 90645484 IC50 = 42.2 nM T64969 CCS47U 90645485 IC50 = 145.2 nM T64969 CXEB69 90645486 IC50 = 102.3 nM T64969 CX29IY 90655145 IC50 = 4 nM T64969 CI56KC 90655146 IC50 > 10000 nM T64969 C5LI2K 90655147 IC50 > 10000 nM T64969 C7J3GQ 90655148 IC50 > 10000 nM T64969 CG09KP 90655149 IC50 = 4997 nM T64969 CJ6EV4 90655150 IC50 > 10000 nM T64969 CE9V5Z 90655151 IC50 = 799 nM T64969 CZ5U8S 90655152 IC50 = 4286 nM T64969 CCFD23 90655153 IC50 = 1699 nM T64969 C3ZFB7 90655154 IC50 = 542 nM T64969 C1NIF5 90655155 IC50 = 3399 nM T64969 C0OIN4 90655156 IC50 = 770 nM T64969 C8O2FA 90655157 IC50 = 6414 nM T64969 CNKM05 90655158 IC50 = 1792 nM T64969 CT7V5Z 90655159 IC50 = 40 nM T64969 CC4M2L 90655160 IC50 = 5 nM T64969 CT4U7R 90655161 IC50 = 1196 nM T64969 CWTH01 90655162 IC50 = 68 nM T64969 C8H7MU 90655163 IC50 = 10 nM T64969 CX2KS1 90655164 IC50 = 20 nM T64969 C5YLC2 90655165 IC50 = 8 nM T64969 CKW2E0 90655166 IC50 = 24 nM T64969 CR9G6B 90655167 IC50 = 8 nM T64969 CW7H2X 90655168 IC50 = 2 nM T64969 CZ2G8V 90655169 IC50 = 139 nM T64969 C3VR8U 90655170 IC50 = 93 nM T64969 C8T9EB 90655171 IC50 = 38 nM T64969 CIW07X 90655172 IC50 = 28 nM T64969 C9D3JH 90655173 IC50 = 4 nM T64969 C8AS4G 90655174 IC50 = 18 nM T64969 CJS7X5 90655175 IC50 = 3 nM T64969 CJ5BC8 90655176 IC50 = 4 nM T64969 CC6BI4 90655177 IC50 = 34 nM T64969 C0ZEA7 90655178 IC50 = 7 nM T64969 CJ6ZX7 90655179 IC50 = 7 nM T64969 CH8QP2 90655180 IC50 = 2159 nM T64969 CI0TR8 90655181 IC50 = 2 nM T64969 CY9FE6 90655275 IC50 = 550 nM T64969 C1CFP6 90655276 IC50 = 575 nM T64969 CI8XW3 90655277 IC50 > 10000 nM T64969 CT28VM 90655278 IC50 > 10000 nM T64969 C8N5TF 90655279 IC50 = 3900 nM T64969 CPN1I6 90655280 IC50 = 1920 nM T64969 CW1LJ4 90655281 IC50 = 43 nM T64969 CAC3D4 90655282 IC50 = 1330 nM T64969 CKO3Z1 90655283 IC50 = 120 nM T64969 C7S8KR 90655284 IC50 = 130 nM T64969 CY0T9O 90655285 IC50 = 43 nM T64969 CG9HX4 90655286 IC50 = 44 nM T64969 C7DT3G 90655287 IC50 = 33 nM T64969 C8RA1Y 90655288 IC50 = 47 nM T64969 C1B7TW 90655289 IC50 = 6 nM T64969 CVO26Z 90655290 IC50 = 5540 nM T64969 CO5M8T 90655291 IC50 = 30 nM T64969 CXNB56 90655292 IC50 > 10000 nM T64969 CW08SL 90655293 IC50 = 680 nM T64969 CC2P7K 90655294 IC50 = 99 nM T64969 CBX47C 90655295 IC50 = 160 nM T64969 CEDA08 90655430 IC50 = 88 nM T64969 C8ZUA3 90655431 IC50 = 877 nM T64969 C82SHX 90655432 IC50 = 184 nM T64969 CEY4A8 90655433 IC50 = 2177 nM T64969 CX5E6G 90655434 IC50 > 10000 nM T64969 COQ34Y 90655435 IC50 = 4706 nM T64969 CPXQ71 90655436 IC50 = 537 nM T64969 C56FLY 90655437 IC50 = 2388 nM T64969 CIQ9S0 90655438 IC50 = 201 nM T64969 C0LFA1 90655439 IC50 = 18020 nM T64969 C3IZ1H 90655440 IC50 = 4150 nM T64969 CT52QD 90655441 IC50 = 32130 nM T64969 C2JX1T 90655442 IC50 = 14700 nM T64969 C2Q1FV 90655443 IC50 = 24050 nM T64969 CR8CQ1 90655444 IC50 = 2090 nM T64969 C4HB6Y 90655445 IC50 = 910 nM T64969 CC76UY 90655446 IC50 = 6150 nM T64969 CC8BR4 90655447 IC50 = 11180 nM T64969 C2BD4K 90655448 IC50 = 1030 nM T64969 C8BL6E 90655679 IC50 = 1580 nM T64969 C2Z7EO 90655680 IC50 = 8660 nM T64969 CAB7E0 90655681 IC50 = 10350 nM T64969 CO8PA3 90655682 IC50 = 7670 nM T64969 C0S1HF 90655767 IC50 > 16000 nM T64969 CW5ZR6 90655768 IC50 = 7670 nM T64969 C51MOA 90655769 IC50 = 3860 nM T64969 CZ6U5W 90655770 IC50 = 1370 nM T64969 C7P6FQ 90655771 IC50 = 84 nM T64969 CXA18Y 90655772 IC50 = 168 nM T64969 C15GJU 90655773 IC50 = 572 nM T64969 C25CWH 90655774 IC50 = 4354 nM T64969 CFRI21 90655775 IC50 = 1201 nM T64969 CAIL45 90655776 IC50 = 1052 nM T64969 CVYA67 90655777 IC50 = 1907 nM T64969 CA84HG 90656352 IC50 = 3960 nM T64969 CW2Z7O 90656353 IC50 = 5530 nM T64969 C0CZ6J 90656354 IC50 = 5260 nM T64969 CRO40H 90656355 IC50 = 650 nM T64969 CQF9S2 90656356 IC50 = 6310 nM T64969 CU12BF 90656357 IC50 = 2800 nM T64969 CO5F7S 90656358 IC50 = 3250 nM T64969 C3PT4O 90656359 IC50 = 120 nM T64969 CP34KC 90664681 IC50 = 1910 nM T64969 CK3IS4 90664930 IC50 = 2280 nM T64969 CRL86F 90665697 IC50 = 650 nM T64969 CR34GP 90666149 IC50 = 9.14 nM T64969 C3RK6C 90666150 IC50 > 1000 nM T64969 CXB1P6 90666151 IC50 = 2.45 nM T64969 CE3VO1 90666152 IC50 = 22.12 nM T64969 C1QYH8 90666153 IC50 = 24.83 nM T64969 C3Q2OD 90666154 IC50 = 10.18 nM T64969 C6CD0G 90666155 IC50 = 77.19 nM T64969 CR1A3V 90666156 IC50 = 6.99 nM T64969 CE6B1Q 90666157 IC50 = 4.68 nM T64969 CP9O1K 90666158 IC50 = 33.95 nM T64969 CSQ89J 90666159 IC50 = 37.37 nM T64969 CF4VN5 90666317 IC50 = 5.78 nM T64969 CNSL72 90666318 IC50 = 6.26 nM T64969 C9V6FU 90666397 IC50 = 520 nM T64969 C5Q8VO 90666398 IC50 = 590 nM T64969 CIB1E8 90666399 IC50 = 570 nM T64969 C08ANK 90666400 IC50 = 800 nM T64969 CL0KH2 90666401 IC50 = 460 nM T64969 C9XI3E 90666402 IC50 = 510 nM T64969 CLF29C 90666403 IC50 > 1000 nM T64969 CU9XB7 90666404 IC50 > 1000 nM T64969 CCL19D 90666405 IC50 > 1000 nM T64969 CYVM38 90666406 IC50 > 1000 nM T64969 CMY4T0 90666407 IC50 > 1000 nM T64969 CNE54X 90666408 IC50 > 1000 nM T64969 CBAM42 90667697 IC50 > 10000 nM T64969 C3TCZ8 90667699 IC50 > 10000 nM T64969 C1M7UL 90667701 IC50 > 10000 nM T64969 C7J0CF 90667703 IC50 > 10000 nM T64969 CU5I7B 90667705 IC50 > 10000 nM T64969 CH16WR 90667707 IC50 > 10000 nM T64969 C8SX2E 90667875 IC50 = 8000 nM T64969 CS73QB 90667877 IC50 = 3900 nM T64969 CSM40E 90667879 IC50 > 10000 nM T64969 CAZD95 90667881 IC50 = 8500 nM T64969 CGU4Q0 90667883 IC50 = 5500 nM T64969 CN1L2V 90667885 IC50 > 10000 nM T64969 C96DTL 90682879 IC50 = 82.3 nM T64969 CF6Q9X 91669170 IC50 = 90 nM T64969 COWV98 91844461 IC50 = 700 nM T64969 C51PJL 91864590 IC50 = 4 nM T64969 C0Y8ZK 91933875 IC50 > 1000 nM T64969 CQTF61 91970514 IC50 = 1600 nM T64969 CE4Q5N 91970515 IC50 = 3900 nM T64969 CC23OD 91970516 IC50 = 900 nM T64969 CB8AR9 91970527 IC50 > 10000 nM T64969 C70ZPT 91971390 Ki = 64 nM T64969 CGQ95X 91971392 Ki = 52 nM T64969 CAU45T 91971978 IC50 > 30000 nM T64969 C64SIO 92042864 IC50 = 409 nM T64969 CWF97Y 92045039 IC50 = 3 nM T64969 C8F7XO 92131166 IC50 = 529.4 nM T64969 CVZ65G 92132732 Ki = 1.5 nM T64969 CMZ92J 92132733 Ki = 1.1 nM T64969 C4CE3S 94146587 IC50 = 34280 nM T64969 CC1Q3Y 95171151 IC50 > 10000 nM T64969 CR02CX 95171152 IC50 = 38 nM T64969 CO4GL7 101879115 IC50 = 0.47 nM T64969 C05NTY 101884761 IC50 = 938000 nM T64969 CWM71R 101884762 IC50 = 600 nM T64969 CRI0S4 101891768 Ki = 12 nM T64969 CK72FW 102129497 IC50 > 10000 nM T64969 CQ7B8D 102515536 Ki = 37 nM T64969 C9SF3U 102515537 Ki = 4 nM T64969 C9G5TC 102515538 Ki = 19 nM T64969 C78NRU 112865697 IC50 = 208 nM T64969 CI6H8C 112865788 IC50 = 974 nM T64969 COU61I 112865858 IC50 = 901 nM T64969 CIR97O 112866175 IC50 = 7.7 nM T64969 C2BAR8 112866205 IC50 = 1188 nM T64969 CU4O5Z 112901888 IC50 = 11000 nM T64969 CM7C3W 117668218 IC50 = 5.9 nM T64969 CTK65N 117668270 IC50 = 208 nM T64969 C63LHQ 117668291 IC50 = 2.2 nM T64969 C0V3ZB 117676956 IC50 < 0.25 nM T64969 CO4Z3X 117676961 IC50 < 0.25 nM T64969 C7RUS2 117676973 IC50 < 0.25 nM T64969 C3NI4J 117676976 IC50 < 0.25 nM T64969 C5LWU4 117677006 IC50 < 0.25 nM T64969 CO01EN 117780037 IC50 = 3 nM T64969 C30HQS 117780120 IC50 = 1860 nM T64969 C2DEK4 117780234 IC50 = 1.5 nM T64969 C5FD2M 117803130 IC50 = 5 nM T64969 CLQ3I0 117803131 IC50 = 6 nM T64969 C21MWK 117803134 IC50 = 2 nM T64969 CX6LJ9 117803651 IC50 = 6 nM T64969 CJYK13 117803656 IC50 = 5 nM T64969 C0MVG2 117803681 IC50 = 20 nM T64969 CXNZ08 117803686 IC50 = 14 nM T64969 CD93GO 117803687 IC50 = 5 nM T64969 CF7O9Z 117803889 IC50 = 9 nM T64969 CW6FL2 118073537 Ki = 9 nM T64969 CBV87I 118073538 Ki = 56 nM T64969 CKX0H7 118073560 IC50 = 1 nM T64969 CKRZ30 118073591 IC50 = 14 nM T64969 C42DMG 118073609 IC50 = 49 nM T64969 CID71C 118073630 IC50 = 194 nM T64969 CEDP63 118073633 IC50 = 6 nM T64969 C1U9WH 118073634 IC50 = 17 nM T64969 C2MDV0 118073642 IC50 = 3 nM T64969 C13PXJ 118073657 IC50 = 29 nM T64969 CGT4R5 118073677 Ki = 2 nM T64969 CMV6T3 118073685 Ki = 152 nM T64969 CKA98U 118073699 IC50 = 387 nM T64969 CUB7S0 118073727 Ki = 6 nM T64969 CLQO21 118073729 IC50 = 4 nM T64969 CVO01M 118073730 Ki = 36 nM T64969 C50FEY 118119835 IC50 = 60 nM T64969 CD8MX0 118223716 IC50 > 50000 nM T64969 CRM37Z 118223719 IC50 = 1.39 nM T64969 C5LNP8 118223723 IC50 > 50000 nM T64969 CB1I5P 118223929 IC50 > 50000 nM T64969 C52ETQ 118223987 IC50 = 16460 nM T64969 CEN18L 118224069 IC50 = 2.18 nM T64969 CTA5U1 118224099 IC50 < 2 nM T64969 CW72PI 118352095 IC50 = 218 nM T64969 CE4NX5 118352096 IC50 = 215 nM T64969 C93WJL 118352106 IC50 = 170 nM T64969 CBNZ41 118352115 IC50 = 80 nM T64969 C7QU3F 118352116 IC50 = 37 nM T64969 CDR52E 118352117 IC50 = 12 nM T64969 C7OUD9 118352135 IC50 = 101 nM T64969 CR7X3L 118352152 IC50 = 17 nM T64969 C2UYT6 118352158 IC50 > 1000 nM T64969 CDWL43 118352163 IC50 > 1000 nM T64969 C8U9AH 118352164 IC50 = 58 nM T64969 CMJ7F6 118352185 IC50 = 266 nM T64969 CQXJ61 118352193 IC50 = 48 nM T64969 CXH1G8 118352197 IC50 = 2 nM T64969 C5O8IG 118352198 IC50 = 192 nM T64969 CH8G4D 118352201 IC50 = 87 nM T64969 CVR8T2 118352210 IC50 = 45 nM T64969 CEM7X4 118352214 IC50 = 22 nM T64969 CC07LP 118352217 IC50 = 128 nM T64969 CAKI19 118514811 IC50 = 5.3 nM T64969 CIY3F2 118578874 IC50 = 287.4 nM T64969 CVHE23 118578939 IC50 = 6 nM T64969 C3D5UB 118661739 Ki = 57 nM T64969 C5Z6CQ 118661749 Ki = 1.1 nM T64969 C5B4MO 118661813 Ki = 34 nM T64969 C4P1SB 118662078 Ki = 44 nM T64969 C15RGE 118692362 IC50 = 20 nM T64969 CIU05O 118710979 IC50 = 10400 nM T64969 CJL49M 118710980 IC50 = 5400 nM T64969 C8WL4B 118710981 IC50 = 18300 nM T64969 C7WCP5 118710982 IC50 = 1100 nM T64969 C8PE2Y 118710983 IC50 = 4300 nM T64969 CBGV74 118710984 IC50 = 1300 nM T64969 CN38JS 118710985 IC50 = 8100 nM T64969 C51LZM 118710986 IC50 = 7000 nM T64969 CU3KJ9 118710987 IC50 = 200 nM T64969 C05DOU 118710988 IC50 = 16700 nM T64969 C4AHL2 118711367 IC50 > 10000 nM T64969 CW8JQ2 118712118 IC50 = 4800 nM T64969 CWO9B7 118715995 IC50 > 100000 nM T64969 C46QUT 118717614 IC50 = 77.2 nM T64969 CJC34Y 118717615 IC50 = 39.2 nM T64969 CFEP93 118717616 IC50 = 28.7 nM T64969 CEC4H0 118717617 IC50 = 89.6 nM T64969 CU2TG3 118717618 IC50 = 92.8 nM T64969 C5OL0W 118717619 IC50 = 110.2 nM T64969 CX0VC6 118719574 IC50 = 16000 nM T64969 C6EX4Q 118719575 IC50 = 6060000 nM T64969 CZEL74 118719576 IC50 = 57000 nM T64969 C01ZDF 118719577 IC50 = 66000 nM T64969 CK01PA 118719578 IC50 = 75000 nM T64969 C4NS1R 118719579 IC50 = 135000 nM T64969 CS3HJ5 118719580 IC50 = 9000000 nM T64969 C3L1TI 118720009 Ki = 28 nM T64969 CI5W9H 118720010 Ki = 14 nM T64969 COQ9S4 118720011 Ki = 18 nM T64969 CV4X8R 118720012 Ki = 114 nM T64969 C5FE8L 118720013 Ki = 423 nM T64969 C7T9VJ 118720014 Ki = 82 nM T64969 CGW7Z0 118721142 IC50 = 3.05 nM T64969 CZJB02 118721143 IC50 = 0.89 nM T64969 CO1B3H 118721144 IC50 = 0.47 nM T64969 C5IVR1 118721145 IC50 = 0.51 nM T64969 CYCQ59 118721146 IC50 = 0.32 nM T64969 CVL8Q3 118721147 IC50 = 0.66 nM T64969 C42NVI 118721148 IC50 = 1.08 nM T64969 C9MKR8 118721149 IC50 = 0.56 nM T64969 C0UA5Q 118721150 IC50 = 0.49 nM T64969 CJS7L9 118721151 IC50 = 0.5 nM T64969 CXHU43 118721152 IC50 = 38.3 nM T64969 CPL9H7 118721153 IC50 = 28.5 nM T64969 C29DWX 118721154 IC50 = 51.2 nM T64969 C9EJO7 118721155 IC50 = 15.1 nM T64969 CB8D5N 118721156 IC50 = 4.9 nM T64969 C5WFB8 118721157 IC50 = 3.43 nM T64969 C0S6RW 118721158 IC50 = 0.53 nM T64969 C20SQV 118721159 IC50 = 1.18 nM T64969 CB9SE1 118722338 IC50 = 2.6 nM T64969 C25AYC 118722339 IC50 = 2.55 nM T64969 CRIG46 118722340 IC50 = 37.9 nM T64969 CA5DI0 118722341 IC50 = 39.2 nM T64969 COB29E 118722342 IC50 = 9.5 nM T64969 CIH6Q8 118722343 IC50 = 11.2 nM T64969 CQ0IG7 118722344 IC50 = 5 nM T64969 C3KLI5 118723185 IC50 > 100000 nM T64969 CJX21C 118724340 IC50 = 0.77 nM T64969 C1C3WP 118724341 IC50 = 0.31 nM T64969 CZC2F3 118724342 IC50 = 0.52 nM T64969 CP9UL3 118724343 IC50 = 1.44 nM T64969 C7UX4R 118724344 IC50 = 0.32 nM T64969 C6Y3VE 118724345 IC50 = 0.65 nM T64969 CEF3I2 118724346 IC50 = 0.26 nM T64969 CW1E0M 118724347 IC50 = 0.57 nM T64969 CZ1G2X 118724348 IC50 = 0.54 nM T64969 CXD08A 118724349 IC50 = 30.5 nM T64969 C3J0KD 118724350 IC50 = 11.9 nM T64969 CY5X0E 118724351 IC50 = 16.6 nM T64969 CUT6Y3 118724352 IC50 = 35.5 nM T64969 CE6Q1K 118724353 IC50 = 20.1 nM T64969 C1J8EN 118724354 IC50 = 0.49 nM T64969 CB8MF7 118724355 IC50 = 0.37 nM T64969 CK28WP 118724356 IC50 = 0.33 nM T64969 CTSC96 118724357 IC50 = 0.78 nM T64969 CZ3LS6 118724358 IC50 = 0.82 nM T64969 C65JUN 118725950 IC50 = 8490 nM T64969 C9HWF5 118726554 IC50 = 1210 nM T64969 C9JKN5 118726555 IC50 = 950 nM T64969 CWYF91 118729842 IC50 = 162.3 nM T64969 CR54XL 118729843 IC50 = 90.3 nM T64969 CF3X9J 118729844 IC50 > 500 nM T64969 CT3Q6C 118729845 IC50 = 298.2 nM T64969 C1QWK6 118729846 IC50 = 226.4 nM T64969 CWUA61 118729847 IC50 = 306.6 nM T64969 C63CDP 118729848 IC50 = 103.2 nM T64969 C1WB7L 118729849 IC50 > 500 nM T64969 C8A7ZT 118729850 IC50 = 3.4 nM T64969 C9WDF4 118729851 IC50 = 102.2 nM T64969 CT08EZ 118729852 IC50 > 500 nM T64969 CG0C5B 118734111 IC50 = 153 nM T64969 COEJ71 118734112 IC50 = 53 nM T64969 CIEY96 118734113 IC50 = 23 nM T64969 CLN1C3 118734114 IC50 > 10000 nM T64969 C4U6AR 118734118 IC50 = 17 nM T64969 CV38ED 118734183 IC50 = 19 nM T64969 C1EI6R 118734184 IC50 = 629 nM T64969 CUJ3W6 118734185 IC50 = 8 nM T64969 CNDX69 118734186 IC50 = 23 nM T64969 CVPH90 118734187 IC50 = 27 nM T64969 CE8WN9 118734188 IC50 = 108 nM T64969 C9M7HI 118734189 IC50 = 275 nM T64969 C7LV4W 118734190 IC50 = 183 nM T64969 CF1ZN3 118734191 IC50 = 241 nM T64969 C7HA2M 118734192 IC50 > 10000 nM T64969 CXB50H 118734193 IC50 = 83 nM T64969 CKZG81 118734194 IC50 = 262 nM T64969 C0W8JD 118734195 IC50 > 10000 nM T64969 C8Y6UI 118734196 IC50 = 183 nM T64969 CMF34Q 118734200 IC50 = 150 nM T64969 CM1KO5 118734202 IC50 = 3883 nM T64969 CA2W7I 118734203 IC50 > 10000 nM T64969 CJ53YU 118734204 IC50 = 7904 nM T64969 C8Q5ZA 118734205 IC50 = 2079 nM T64969 CXW73G 118734207 IC50 = 1374 nM T64969 C6J8NH 118734208 IC50 = 415 nM T64969 C16HCZ 118734209 IC50 = 80 nM T64969 COI6J1 118734210 IC50 = 170 nM T64969 C45FIB 118734211 IC50 = 55 nM T64969 CLC85D 118734212 IC50 = 173 nM T64969 CC9S3Y 118734213 IC50 = 5 nM T64969 CG0JF1 118734214 IC50 = 18 nM T64969 CRQ98M 118734215 IC50 = 220 nM T64969 CY7ES4 118736528 IC50 = 7000 nM T64969 CT16XS 118736529 IC50 = 4800 nM T64969 CWNC90 118736530 IC50 > 10000 nM T64969 C8OP4R 118736531 IC50 > 10000 nM T64969 C75QPF 118736532 IC50 > 10000 nM T64969 CV9DL6 118736533 IC50 > 10000 nM T64969 C2VOS9 118736534 IC50 = 8700 nM T64969 CD4ZL0 118736535 IC50 > 10000 nM T64969 C18AYF 118736536 IC50 > 10000 nM T64969 CWI2O0 118736537 IC50 = 7200 nM T64969 C8HLE3 118736538 IC50 > 10000 nM T64969 CNTP03 118736539 IC50 > 10000 nM T64969 CYP1V5 118736540 IC50 > 10000 nM T64969 CMEK38 118736541 IC50 > 10000 nM T64969 C7EJ4B 118736542 IC50 > 10000 nM T64969 CU8D2K 118736543 IC50 > 10000 nM T64969 CAO94Z 118736544 IC50 = 3270 nM T64969 CCX29A 118736545 IC50 = 5600 nM T64969 CLI75H 118736546 IC50 > 10000 nM T64969 CQCX41 118737057 IC50 = 3518 nM T64969 CDBZ85 118738351 IC50 = 26 nM T64969 CJV62R 118738352 IC50 = 12.5 nM T64969 CSTB45 118738353 IC50 = 10.8 nM T64969 CM38XC 118738354 IC50 = 28 nM T64969 C1EDA6 118738355 IC50 = 59.9 nM T64969 C63SVY 118738356 IC50 = 11.4 nM T64969 CQ83JA 118738357 IC50 = 232.4 nM T64969 CUY8Z3 118900244 IC50 = 2.84 nM T64969 CB85RT 118900245 IC50 = 1.54 nM T64969 CR2X9A 118900269 IC50 = 153.5 nM T64969 CH3I9B 118900282 IC50 = 0.76 nM T64969 CI3TK4 118900289 IC50 = 1.48 nM T64969 C7V3DH 118900298 IC50 = 0.69 nM T64969 C0LIS1 118900305 IC50 = 0.94 nM T64969 CINT13 118900306 IC50 = 2.73 nM T64969 C9ARH1 118912888 IC50 = 6 nM T64969 CON03D 121231412 IC50 = 3 nM T64969 CBRZ51 121280156 IC50 > 600 nM T64969 CRQ3I6 121396150 IC50 = 11 nM T64969 CILM06 121423933 IC50 = 31 nM T64969 CN5CA4 121427628 IC50 = 5 nM T64969 CWA94G 122182409 IC50 > 100000 nM T64969 C02HIB 122186131 IC50 = 1100 nM T64969 C75JDA 122186132 IC50 = 100 nM T64969 CHG54X 122186133 IC50 > 10000 nM T64969 CS02EL 122186134 IC50 > 10000 nM T64969 CI35QX 122186135 IC50 = 400 nM T64969 C6PGI7 122186136 IC50 > 10000 nM T64969 CDKC89 122186137 IC50 = 300 nM T64969 CRH7T4 122186138 IC50 > 10000 nM T64969 CPO72V 122186139 IC50 = 2500 nM T64969 C56DAE 122186140 IC50 = 2100 nM T64969 CM5FZ6 122186141 Ki = 0.64 nM T64969 C98PCS 122186142 IC50 > 10000 nM T64969 C7R1JK 122186143 IC50 = 4900 nM T64969 CQCM53 122186144 IC50 = 1400 nM T64969 CS4LP5 122186145 IC50 = 900 nM T64969 C4VM5U 122186146 IC50 > 10000 nM T64969 C8VBX6 122186147 IC50 = 1900 nM T64969 CT9M5F 122186148 IC50 > 10000 nM T64969 CPD83K 122186149 IC50 = 1500 nM T64969 CA3SU2 122186150 Ki = 0.32 nM T64969 CI8RS6 122186151 IC50 = 8600 nM T64969 CU04WQ 122186152 IC50 = 700 nM T64969 C8DY3H 122186153 IC50 = 300 nM T64969 COMH39 122186154 IC50 = 3600 nM T64969 CTXU80 122186155 IC50 = 4900 nM T64969 C4P0JT 122188303 IC50 = 470 nM T64969 CSR50M 122188304 IC50 = 190 nM T64969 CRUV12 122188305 IC50 = 26 nM T64969 C6U3ER 122188306 IC50 = 5100 nM T64969 C3WB0T 122188307 IC50 > 10000 nM T64969 C3WLR4 122188308 IC50 > 10000 nM T64969 CMZX95 122188309 IC50 = 340 nM T64969 CC3BG6 122188310 IC50 > 10000 nM T64969 C57DPM 122188311 IC50 > 10000 nM T64969 C30MSH 122188312 IC50 = 560 nM T64969 C2F1DC 122188313 IC50 = 1300 nM T64969 CP8IB7 122188314 IC50 = 5500 nM T64969 C0C8EB 122188315 IC50 = 440 nM T64969 CEK54V 122188316 IC50 = 7800 nM T64969 C4S5QU 122188317 IC50 = 5700 nM T64969 C2H1AO 122188318 IC50 > 10000 nM T64969 C0VIM6 122188319 IC50 > 10000 nM T64969 C0D2EB 122188320 IC50 = 1200 nM T64969 C64GES 122188321 IC50 > 10000 nM T64969 C7GV9B 122188322 IC50 = 7500 nM T64969 C2LBT7 122188323 IC50 > 10000 nM T64969 C0ZIQ6 122188324 IC50 > 10000 nM T64969 CW3Q5T 122188325 IC50 > 10000 nM T64969 CKU2O7 122188326 IC50 > 10000 nM T64969 CS3Z2X 122188327 IC50 = 780 nM T64969 CFO57L 122188328 IC50 > 10000 nM T64969 CNF7Q2 122188329 IC50 = 7.3 nM T64969 C7RU0L 122188330 IC50 > 10000 nM T64969 CGZJ16 122188331 IC50 > 10000 nM T64969 C8O7SU 122188332 IC50 = 130 nM T64969 C8G4QO 122188333 IC50 = 2300 nM T64969 CO96BU 122188334 IC50 = 140 nM T64969 C0HBC8 122188335 IC50 = 53 nM T64969 C79UWR 122188336 IC50 = 20 nM T64969 CCP8B1 122188337 IC50 = 8.7 nM T64969 C4BOF5 122188338 IC50 = 160 nM T64969 CAS18Q 122188339 IC50 > 10000 nM T64969 CYPA94 122188340 IC50 > 10000 nM T64969 C52ERC 122188341 IC50 = 660 nM T64969 CYW1M5 122188342 IC50 = 1500 nM T64969 CCV6T9 122189237 IC50 = 5283 nM T64969 C61RXE 122189241 IC50 = 4824 nM T64969 CG7P6E 122189248 IC50 = 0.037 nM T64969 C0YZ4K 122191926 IC50 > 1000 nM T64969 C6Q5CB 122191927 IC50 = 1.2 nM T64969 CZG10A 122191928 IC50 = 573.6 nM T64969 CB9XO4 122191929 IC50 = 102.3 nM T64969 C7R8AM 122191930 IC50 > 1000 nM T64969 C2GP3K 122191931 IC50 = 5.4 nM T64969 CH0J8K 122191932 IC50 = 1.2 nM T64969 CM8G5F 122191933 IC50 = 3 nM T64969 CZB2R1 122191934 IC50 = 510.2 nM T64969 CO43WT 122191935 IC50 = 133.9 nM T64969 CB3FU0 122191936 IC50 = 9 nM T64969 CVEQ28 122191937 IC50 > 1000 nM T64969 C8YIT6 122191938 IC50 = 147.4 nM T64969 C31QLD 122191939 IC50 = 26.9 nM T64969 C1JQ0L 122191940 IC50 = 8.9 nM T64969 C6CGK1 122191941 IC50 = 5.5 nM T64969 C0SAT2 122191942 IC50 > 1000 nM T64969 C4M3OA 122191943 IC50 > 1000 nM T64969 CB8DC6 122191944 IC50 > 1000 nM T64969 CZFO12 122191945 IC50 > 1000 nM T64969 C7YZE5 122191946 IC50 > 1000 nM T64969 C7NV0K 122191947 IC50 > 1000 nM T64969 CPK50T 122191948 IC50 = 0.9 nM T64969 CF4E8L 122191949 IC50 = 2.1 nM T64969 CTI7K9 122191950 IC50 = 6.5 nM T64969 C83TUO 122191951 IC50 = 9.6 nM T64969 CFS29N 122191952 IC50 = 6.9 nM T64969 C25QVG 122191953 IC50 = 141 nM T64969 C5O8VS 122191954 IC50 = 7 nM T64969 CY24OJ 122191955 IC50 = 5.3 nM T64969 C2A9MG 122191956 IC50 = 3.3 nM T64969 CVT7W4 122191957 IC50 = 2.4 nM T64969 CRM0T2 122191958 IC50 = 5.6 nM T64969 C8ZPL5 122191959 IC50 = 7.9 nM T64969 CNU1X5 122191960 IC50 = 4.2 nM T64969 CL8M2N 122191961 IC50 = 6.4 nM T64969 C4X7SD 122192466 IC50 > 10000 nM T64969 CJ6RO8 122193596 IC50 > 10000 nM T64969 CB6M4T 122193759 IC50 > 10000 nM T64969 C65XUZ 122193760 IC50 > 10000 nM T64969 CHF47Y 122193761 IC50 > 10000 nM T64969 C1XHI4 122193762 IC50 = 7710 nM T64969 CNX0Q2 122193763 IC50 > 10000 nM T64969 CWV0C3 122193764 IC50 > 10000 nM T64969 CSG98Y 122193765 IC50 = 3950 nM T64969 C1SED2 122193766 IC50 > 10000 nM T64969 CINA05 122193767 IC50 > 10000 nM T64969 C27WGV 122193768 IC50 > 10000 nM T64969 CCLQ75 122193769 IC50 > 10000 nM T64969 CXDR48 122193770 IC50 > 10000 nM T64969 C96LDU 122193771 IC50 > 10000 nM T64969 C50HEA 122193772 IC50 > 10000 nM T64969 CPA8C5 122193773 IC50 > 10000 nM T64969 C83XVM 122193778 IC50 = 21180 nM T64969 CIS0B2 122193779 IC50 = 21560 nM T64969 C26POY 122193780 IC50 = 45700 nM T64969 C59RDU 122193840 IC50 = 3290 nM T64969 CXE87R 122193841 IC50 = 1260 nM T64969 CM8N1W 122195059 IC50 = 348 nM T64969 CC5KB6 122195541 IC50 = 4 nM T64969 CKG14J 122195542 IC50 = 543 nM T64969 CIPZ05 122195677 IC50 = 186 nM T64969 C4V5WK 122195678 IC50 = 29 nM T64969 C03XJB 122195679 IC50 > 10000 nM T64969 C2CM8S 122195680 IC50 = 35 nM T64969 CIC6N1 122195681 IC50 = 227 nM T64969 C3F1YP 122195682 IC50 = 23 nM T64969 C4IMA2 122195683 IC50 > 10000 nM T64969 C8TK1W 122195684 IC50 = 812 nM T64969 C4FXV5 122195685 IC50 = 1020 nM T64969 C47QYW 122195686 IC50 > 10000 nM T64969 CZC4K1 122195687 IC50 = 445 nM T64969 CK0Q3A 122195688 IC50 = 3050 nM T64969 CLTG90 122195689 IC50 = 9 nM T64969 C0TX3A 122195690 IC50 = 31 nM T64969 C52BMS 122195691 IC50 = 1460 nM T64969 C1KXL8 122205446 IC50 = 280 nM T64969 C4XIQ7 122205447 IC50 = 21 nM T64969 C3BL8I 122205448 IC50 > 1000 nM T64969 C37ICD 122417697 IC50 = 363.3 nM T64969 C9D5RK 122417700 IC50 = 57.8 nM T64969 CQD76R 122417702 IC50 = 76.1 nM T64969 C47VHI 122417706 IC50 = 6.7 nM T64969 CBF3G5 122417707 IC50 = 10.9 nM T64969 C69PHO 122417709 IC50 = 3.6 nM T64969 CW64ZC 122417712 IC50 = 53.1 nM T64969 C5BMI1 122417713 IC50 > 1000 nM T64969 C1YRN4 122417718 IC50 = 82.5 nM T64969 CE45KB 122417721 IC50 = 416.1 nM T64969 C9LK2Y 122417722 IC50 > 1000 nM T64969 C5RD4P 122417724 IC50 = 232.3 nM T64969 CAG29M 122417725 IC50 = 351.8 nM T64969 C6QMU4 122417730 IC50 = 16.7 nM T64969 C90XRZ 122417735 IC50 = 8.1 nM T64969 CFSK74 122417740 IC50 > 1000 nM T64969 CWT4F3 122417747 IC50 = 102.6 nM T64969 CHY1Z0 122417753 IC50 > 1000 nM T64969 CC04MJ 122417757 IC50 = 46.28 nM T64969 C35XVJ 122417762 IC50 = 43.8 nM T64969 C9WJ6T 122417763 IC50 = 36.2 nM T64969 C19SAP 122417767 IC50 = 9.2 nM T64969 C1VP7E 122417768 IC50 = 22.5 nM T64969 CV68FJ 122417770 IC50 = 27.3 nM T64969 CIG7Y6 122417773 IC50 > 1000 nM T64969 CD37VR 122417777 IC50 = 10.5 nM T64969 C0IJR1 122417781 IC50 = 4.4 nM T64969 C0XFJ2 122417784 IC50 = 24.1 nM T64969 C4LV6K 122417787 IC50 = 162.7 nM T64969 C2VP7F 122417788 IC50 = 139 nM T64969 C8UF2Q 122417837 IC50 = 184.5 nM T64969 C6DAO2 122417839 IC50 = 313.6 nM T64969 CDT5O1 122417840 IC50 = 23.7 nM T64969 CJ6D9N 122417841 IC50 = 74.6 nM T64969 CAM13U 122417842 IC50 = 387.8 nM T64969 CFL0M8 122417848 IC50 > 1000 nM T64969 C1TIR7 122417852 IC50 = 247.2 nM T64969 CWL2N6 122417856 IC50 = 109.1 nM T64969 C9VTO7 122417858 IC50 = 2 nM T64969 C9QB1R 122417864 IC50 = 9.7 nM T64969 C6QHB4 122484585 IC50 = 0.3 nM T64969 CRT93E 122484586 IC50 = 1.2 nM T64969 CF7ME6 122484587 IC50 = 16 nM T64969 CX8EC3 122484589 IC50 = 111 nM T64969 C2E8NC 122484594 IC50 = 14 nM T64969 CJ63LF 122484678 IC50 = 70 nM T64969 C6DP2N 122484680 IC50 = 68 nM T64969 C2SXK9 122484682 IC50 = 314 nM T64969 C8MJ4P 122484684 IC50 = 180 nM T64969 C1U2WJ 122484694 IC50 = 0.4 nM T64969 CJC73G 122484695 IC50 = 3.8 nM T64969 C4AUD3 122484700 IC50 = 0.8 nM T64969 CS58YZ 122484702 IC50 = 30 nM T64969 CX6KW7 122484733 IC50 = 115 nM T64969 CV63PN 122484734 IC50 = 1 nM T64969 C1NPL5 122484735 IC50 = 6.8 nM T64969 C01SPL 122484737 IC50 = 0.7 nM T64969 CLM7K3 122604539 IC50 > 10000 nM T64969 C01JHI 122604566 IC50 > 10000 nM T64969 CIR1B3 123134714 IC50 = 2.4 nM T64969 CY30FL 123752658 IC50 > 100 nM T64969 CZAY93 124197376 IC50 = 4.1 nM T64969 C5T9NG 124197380 IC50 = 5 nM T64969 CZFG57 124197588 IC50 = 8.4 nM T64969 CH0B7X 124222449 Ki = 161 nM T64969 CIP4Q6 124435382 IC50 = 147 nM T64969 CAXY02 125461985 IC50 = 2 nM T64969 CCX79B 126667178 IC50 = 2100 nM T64969 C97OIS 127024859 IC50 = 21 nM T64969 CBU92A 127024861 IC50 = 7 nM T64969 CJB02T 127024862 IC50 = 0.5 nM T64969 C5P6VB 127024863 IC50 = 4 nM T64969 CEI65V 127024864 IC50 = 0.4 nM T64969 CIB0W9 127024865 IC50 = 3 nM T64969 CE89QB 127024882 IC50 > 10000 nM T64969 CUF81C 127025156 IC50 > 500 nM T64969 CP3LK5 127025157 IC50 = 14.83 nM T64969 C8QKX6 127025158 IC50 = 97.22 nM T64969 C86RIQ 127025203 IC50 = 300 nM T64969 CDQ52G 127025443 IC50 = 48.81 nM T64969 CZH1K2 127025487 Ki > 2000 nM T64969 COA80E 127025789 IC50 = 2 nM T64969 CL4YH3 127025790 IC50 = 0.9 nM T64969 CYQ2U3 127025791 IC50 = 2 nM T64969 CZRI81 127025792 IC50 = 21 nM T64969 C8KXV1 127025843 IC50 > 1000 nM T64969 CG3T9I 127026061 IC50 = 6 nM T64969 CVYD73 127026080 IC50 = 0.9 nM T64969 C27YJQ 127026081 IC50 = 2 nM T64969 CFV5O3 127026082 IC50 = 1.5 nM T64969 CGT0I1 127026385 Ki = 10.4 nM T64969 CQ8EW1 127026406 IC50 = 9 nM T64969 CW6PB1 127026407 IC50 = 3 nM T64969 CVRP85 127026408 IC50 = 20 nM T64969 C3Y0XF 127026464 IC50 = 5 nM T64969 C1V2ZA 127026465 IC50 = 19 nM T64969 C7A4QX 127026466 IC50 = 7 nM T64969 CCI6J7 127026467 IC50 = 41 nM T64969 CEM1T3 127026690 IC50 = 276 nM T64969 CI3HN6 127026710 IC50 = 0.5 nM T64969 CY1K9D 127027073 IC50 = 48 nM T64969 C41EAT 127027074 IC50 = 5 nM T64969 CBA80X 127027086 IC50 = 13 nM T64969 CWK63L 127027087 IC50 = 59 nM T64969 CRQ0E7 127027088 IC50 = 8 nM T64969 CV34HC 127027089 IC50 = 5 nM T64969 CIKQ57 127027090 IC50 = 26 nM T64969 CBT52X 127027296 IC50 = 66.59 nM T64969 CS6TJ8 127027297 IC50 = 90.57 nM T64969 C0EZA2 127027298 IC50 > 500 nM T64969 CER0Q3 127027305 IC50 = 78.17 nM T64969 CAH9J6 127027306 IC50 = 476.66 nM T64969 CN3SW5 127027307 IC50 = 71.82 nM T64969 CC0R4L 127027308 IC50 = 121.09 nM T64969 C9E7CQ 127027332 IC50 > 10000 nM T64969 CA59WC 127027333 IC50 = 730 nM T64969 CQXW85 127027334 IC50 > 10000 nM T64969 CPLE01 127027335 IC50 > 10000 nM T64969 CSM76Y 127027336 IC50 > 10000 nM T64969 C7EYC2 127027620 IC50 = 26.56 nM T64969 C12ODR 127027621 IC50 = 131.09 nM T64969 CA7JW5 127027622 IC50 = 455.17 nM T64969 CMT3C7 127027623 IC50 = 290.46 nM T64969 C0T3HO 127027641 IC50 = 495.3 nM T64969 CLO6P4 127027642 IC50 = 165.6 nM T64969 C14WBS 127027666 IC50 = 8 nM T64969 CUG53Q 127027694 Ki = 0.6 nM T64969 CE1BH6 127027695 Ki = 844 nM T64969 CM2S6K 127027696 Ki = 389 nM T64969 CRZA23 127027741 IC50 = 159 nM T64969 CV7R6H 127027985 IC50 = 2 nM T64969 C0Q6RG 127027992 IC50 = 130 nM T64969 CO3P6I 127028013 Ki > 2000 nM T64969 C3O4AR 127028014 Ki = 3 nM T64969 C1A3FO 127028015 Ki = 2 nM T64969 CG7ZB1 127028016 Ki = 8 nM T64969 CW5EY8 127028017 Ki = 17 nM T64969 CE62DA 127028049 IC50 = 4.52 nM T64969 C0HAR2 127028050 IC50 = 2.92 nM T64969 C82RGS 127028051 IC50 = 10.8 nM T64969 C7SIV9 127028052 IC50 = 5.01 nM T64969 CH1TO3 127028299 Ki = 134 nM T64969 C04MHS 127028310 IC50 = 150 nM T64969 C85ZEY 127028311 IC50 = 20 nM T64969 C5V3SU 127028312 IC50 = 1330 nM T64969 C6C0QK 127028313 IC50 = 690 nM T64969 CXE58H 127028337 Ki = 17 nM T64969 CZK9V1 127028338 Ki = 747 nM T64969 CG7I9K 127028339 Ki > 2000 nM T64969 CIZ7M1 127028340 Ki > 2000 nM T64969 C43XYB 127028671 Ki = 22.4 nM T64969 CG9M4V 127028672 Ki = 4 nM T64969 CI7TC8 127028673 Ki = 16 nM T64969 CR9A4B 127028681 Ki = 57 nM T64969 CK71GH 127028959 Ki = 6.5 nM T64969 C9XH6D 127028969 IC50 = 1110 nM T64969 C9CMQ6 127028970 IC50 = 4610 nM T64969 CXFB96 127028971 IC50 > 10000 nM T64969 CYAT13 127028990 Ki = 519 nM T64969 C4QX6U 127028991 Ki = 85 nM T64969 CVR5S1 127028992 Ki = 104 nM T64969 C4Y8CR 127028993 Ki = 732 nM T64969 CFN3D7 127028994 Ki = 5.6 nM T64969 CLK2Z3 127028995 Ki = 175 nM T64969 C64UOV 127029263 IC50 = 760 nM T64969 C69BON 127029520 IC50 = 13 nM T64969 C1XD6R 127029809 IC50 > 100000 nM T64969 CI1E5W 127029864 IC50 = 582.17 nM T64969 C9CDQ5 127029901 IC50 = 434.1 nM T64969 C4I7ZN 127029902 IC50 = 353.7 nM T64969 CHPZ40 127029903 IC50 = 823.9 nM T64969 C4KF0T 127030085 Ki = 15 nM T64969 CG2DM3 127030086 Ki = 32 nM T64969 CTA3J6 127030119 Ki = 346 nM T64969 CO0I4A 127030120 Ki = 82 nM T64969 C4WY3P 127030121 Ki = 155 nM T64969 C6PK2L 127030122 Ki = 629 nM T64969 CVBF01 127030212 IC50 > 10000 nM T64969 CI93ZA 127030213 IC50 > 10000 nM T64969 C70DZQ 127030241 IC50 = 594.5 nM T64969 C1D8OL 127030242 IC50 = 518.6 nM T64969 C60QMN 127030384 Ki = 10 nM T64969 C8LQV4 127030516 IC50 > 10000 nM T64969 CV2EA7 127030757 Ki > 2060 nM T64969 CT7SX1 127031071 Ki = 108 nM T64969 C4U1NV 127031072 Ki = 95 nM T64969 CD4RB2 127031073 Ki = 145 nM T64969 CL31XR 127031074 Ki > 688 nM T64969 C0BR2L 127031164 IC50 = 89.6 nM T64969 CN9IV4 127031165 IC50 = 186.9 nM T64969 C2O1VX 127031166 IC50 = 829.2 nM T64969 CS12RU 127031435 IC50 > 10000 nM T64969 CZXP62 127031750 IC50 > 10000 nM T64969 CD45KQ 127031941 Ki = 61 nM T64969 C3E5YO 127032014 IC50 > 10000 nM T64969 C2ZD8S 127032024 IC50 > 10000 nM T64969 CXWY73 127032324 IC50 > 10000 nM T64969 C42UOD 127032352 IC50 = 245.1 nM T64969 CV42MI 127032353 IC50 = 63.1 nM T64969 CJ59GA 127032541 Ki = 330 nM T64969 CS40XR 127032999 IC50 = 137.9 nM T64969 CQ1I3B 127033227 Ki = 37 nM T64969 C59MVH 127033228 Ki > 2060 nM T64969 CR2P3O 127033504 Ki = 51 nM T64969 CB35SE 127033505 Ki = 15 nM T64969 C2GLU3 127033506 Ki = 12 nM T64969 C81SKW 127033507 Ki = 78 nM T64969 C46AWH 127033508 Ki = 26 nM T64969 CWIO91 127033509 Ki = 31 nM T64969 CJZT54 127033800 Ki = 625 nM T64969 CL7P4Q 127033902 Ki = 590 nM T64969 C9BYR7 127034155 IC50 = 460 nM T64969 CL67CH 127034156 IC50 = 115.9 nM T64969 C3ZTY9 127034157 IC50 = 99 nM T64969 C5EM4W 127034158 IC50 = 456.2 nM T64969 C97FGP 127034305 Ki = 349 nM T64969 C52FRX 127034424 IC50 = 211.4 nM T64969 CEDK31 127034582 Ki = 144 nM T64969 CKS28E 127034802 IC50 = 350 nM T64969 CWRB15 127034986 IC50 = 71.71 nM T64969 CM09WL 127035009 IC50 = 18.04 nM T64969 CDU87A 127035163 IC50 = 94.82 nM T64969 CPN2Q6 127035597 Ki = 196 nM T64969 CEPL09 127036182 IC50 = 310.76 nM T64969 C87BIU 127036183 IC50 = 102.93 nM T64969 CR0NI6 127036477 IC50 = 317.12 nM T64969 CM17TO 127036596 IC50 = 24.81 nM T64969 C3SPE9 127036731 Ki = 7.4 nM T64969 CGOK31 127036732 Ki = 9.5 nM T64969 C52JBY 127036758 IC50 = 362 nM T64969 C72EXH 127036764 IC50 = 189.49 nM T64969 CKX40V 127037812 IC50 > 10000 nM T64969 C93RQT 127038361 IC50 = 9190 nM T64969 CHMT84 127038362 IC50 = 4480 nM T64969 CVU8Z4 127038363 IC50 = 3220 nM T64969 CB73NS 127038364 IC50 = 7880 nM T64969 C70RUP 127038480 IC50 > 10000 nM T64969 CEG89U 127038628 IC50 = 25580 nM T64969 CJHQ62 127038729 IC50 = 3200 nM T64969 CSV0T8 127039237 IC50 = 9.1 nM T64969 C18SAK 127039275 IC50 = 4130 nM T64969 C5GJ1F 127039276 IC50 = 5960 nM T64969 CYNR48 127039277 IC50 = 301.3 nM T64969 CLI54D 127039495 IC50 = 1680 nM T64969 C03PVF 127039496 IC50 = 2270 nM T64969 CRS60P 127039497 IC50 = 5670 nM T64969 C4BY1V 127039518 IC50 = 11570 nM T64969 C87AFX 127039599 IC50 = 6683.44 nM T64969 CUVR09 127039608 IC50 = 8540 nM T64969 COE17A 127039609 IC50 = 21310 nM T64969 C93XHQ 127039610 IC50 = 9594.01 nM T64969 CXLQ81 127039662 IC50 = 12240 nM T64969 CW4S0U 127039718 IC50 = 3890 nM T64969 C8BSO6 127039719 IC50 = 5430 nM T64969 CNH94T 127039720 IC50 = 2550 nM T64969 C01LGZ 127039804 IC50 = 4670 nM T64969 CO4N6V 127039812 IC50 = 790 nM T64969 CEU27C 127039813 IC50 = 2350 nM T64969 C48BVH 127039814 IC50 = 720 nM T64969 CBM41V 127039833 IC50 = 790 nM T64969 C91FAK 127039834 IC50 = 680 nM T64969 C6OU4T 127039835 IC50 = 2520 nM T64969 C3N2YV 127039870 IC50 = 3.6 nM T64969 CKT2I9 127039915 IC50 = 26920 nM T64969 CEQA86 127039935 IC50 = 600 nM T64969 CTK6W3 127039936 IC50 = 1450 nM T64969 CB3X9Y 127039944 IC50 = 15160 nM T64969 CAL3D1 127039945 IC50 = 7379.04 nM T64969 CB5KT1 127039946 IC50 = 9260 nM T64969 C03XGE 127040180 IC50 = 2380 nM T64969 C7CNB9 127040181 IC50 = 4320 nM T64969 C8PK1U 127040288 IC50 = 5023.43 nM T64969 CT4U6D 127040940 IC50 = 6580 nM T64969 CJ8E7C 127040941 IC50 = 1260 nM T64969 CA6RH0 127040942 IC50 = 10690 nM T64969 CP6D1T 127040943 IC50 = 10939.56 nM T64969 CYM0T6 127041396 IC50 = 3560 nM T64969 CXM5Q6 127041397 IC50 = 4490 nM T64969 CJI9D7 127041398 IC50 = 3780 nM T64969 CGX1C5 127041399 IC50 = 2560 nM T64969 C6Z5KQ 127041488 IC50 = 860 nM T64969 C3WCN8 127041777 IC50 > 10000 nM T64969 CV53TB 127041787 IC50 = 1510 nM T64969 CP03MA 127042285 IC50 = 1.12 nM T64969 C4M7QX 127042286 IC50 = 15.4 nM T64969 CK5H8B 127042641 IC50 = 2.01 nM T64969 CNA9F0 127042642 IC50 = 4.62 nM T64969 CQNL56 127042643 IC50 = 4.71 nM T64969 C5PFK0 127042644 IC50 = 6.02 nM T64969 C1G9QI 127042685 IC50 = 2890 nM T64969 CZ3J4V 127042686 IC50 = 3670 nM T64969 C27XTM 127042687 IC50 = 5100 nM T64969 CUY35P 127042939 IC50 = 1.63 nM T64969 CP15ZX 127043295 IC50 = 2.97 nM T64969 C1ID2U 127044206 IC50 = 880 nM T64969 CV0F3N 127045112 IC50 = 28.2 nM T64969 CTPY32 127045266 IC50 = 44.1 nM T64969 CWI8Q2 127045267 IC50 = 3.58 nM T64969 CV5I8S 127045270 IC50 = 31.9 nM T64969 CL9BQ0 127045740 IC50 = 4.4 nM T64969 CG1OT5 127045741 IC50 = 38.8 nM T64969 C3M7AZ 127045742 IC50 = 3.7 nM T64969 CHK16Q 127045929 IC50 > 1000 nM T64969 CG70DF 127046321 IC50 = 0.4 nM T64969 CHT3M0 127046322 IC50 = 0.7 nM T64969 C3R7UG 127046487 IC50 = 7.3 nM T64969 CRWO38 127046488 IC50 = 1.8 nM T64969 CAK4O6 127046533 IC50 = 3.6 nM T64969 CZ6A2F 127046534 IC50 = 5.8 nM T64969 CO4N3J 127047042 IC50 = 49000 nM T64969 CL18YE 127047185 IC50 = 34000 nM T64969 C8TIY1 127047186 IC50 = 35000 nM T64969 CVC5W1 127047187 IC50 = 15000 nM T64969 CW5X1G 127047188 IC50 = 38000 nM T64969 CO96WN 127047445 IC50 = 9.6 nM T64969 CY3J0C 127047591 IC50 > 1000 nM T64969 C81WZQ 127048296 IC50 = 259 nM T64969 CDL7Z4 127048297 IC50 > 500 nM T64969 CGXU78 127048860 IC50 = 20.5 nM T64969 C7Q0FC 127048861 IC50 = 58.8 nM T64969 C0V7YZ 127048976 IC50 = 2.04 nM T64969 CMTG09 127048977 IC50 = 0.854 nM T64969 CDWM04 127048978 IC50 = 0.662 nM T64969 CPH4B3 127048979 IC50 = 3.96 nM T64969 CN1WT6 127048980 IC50 = 1.43 nM T64969 CQ83OB 127048981 IC50 = 0.772 nM T64969 CAY75H 127048991 EC50 = 360 nM T64969 C8M1LU 127049195 IC50 = 25.86 nM T64969 C4X2CJ 127049305 EC50 = 1780 nM T64969 CVZE82 127049306 EC50 = 18 nM T64969 C5ZF0X 127049307 EC50 = 150 nM T64969 CAX68G 127049308 EC50 = 10 nM T64969 CR64FG 127049380 IC50 = 1.34 nM T64969 CLF41Y 127049383 IC50 = 5.52 nM T64969 CVH72U 127049689 IC50 = 0.803 nM T64969 CP2NO1 127049690 IC50 = 194 nM T64969 C6A2IV 127050067 IC50 = 1.98 nM T64969 C1TAI8 127050068 IC50 = 294.6 nM T64969 CIV53M 127050256 EC50 = 22 nM T64969 C82WZB 127050549 EC50 = 1340 nM T64969 C16LRJ 127050550 EC50 = 390 nM T64969 CR3KX5 127050551 EC50 > 20000 nM T64969 C95CNQ 127050554 IC50 = 5.06 nM T64969 C1PFS7 127050555 IC50 = 247 nM T64969 CJ5L8A 127050556 IC50 < 0.495 nM T64969 CB3G8V 127050557 IC50 = 1.5 nM T64969 CYT6X9 127050558 EC50 = 24 nM T64969 C1PHY6 127050559 EC50 = 15 nM T64969 C8I2MC 127050881 EC50 = 550 nM T64969 CJ4WY0 127050882 EC50 = 7 nM T64969 CBS36H 127051046 IC50 = 200.3 nM T64969 CE7B3D 127051146 IC50 = 200 nM T64969 C6XHP2 127051445 IC50 < 1 nM T64969 CO29UV 127051446 EC50 > 30000 nM T64969 CQW87Z 127051447 EC50 = 73 nM T64969 CX31ZJ 127051448 EC50 = 23 nM T64969 CD0CG5 127051556 IC50 = 25.53 nM T64969 CHF7B5 127051692 IC50 = 9040 nM T64969 C4KLU2 127051866 IC50 = 4.54 nM T64969 CI9Y4N 127051867 IC50 = 1.19 nM T64969 CH4AJ8 127052082 EC50 = 14900 nM T64969 C7V9BT 127052091 IC50 = 2.25 nM T64969 CHQG07 127052092 IC50 = 80 nM T64969 C9XM4K 127052093 IC50 = 2.26 nM T64969 CSO2J4 127052094 EC50 = 12 nM T64969 C1AK9H 127052095 EC50 = 24 nM T64969 CQG69I 127052096 EC50 = 15 nM T64969 CH51IT 127052097 EC50 = 9 nM T64969 C5N0QK 127052408 IC50 = 296 nM T64969 CO3E8G 127052409 IC50 = 9.05 nM T64969 CB5YE2 127052414 EC50 = 14 nM T64969 CZ52FH 127052605 IC50 = 18.48 nM T64969 C0D6UI 127052606 IC50 = 21.95 nM T64969 CSM21N 127052640 IC50 = 192000 nM T64969 CN6V5E 127052874 IC50 > 300000 nM T64969 C1T8EL 127052875 IC50 > 300000 nM T64969 CUO7X0 127052876 IC50 = 7920 nM T64969 CGKZ89 127052877 IC50 = 81200 nM T64969 C1PK0X 127052898 IC50 = 83.88 nM T64969 CZ37CP 127052899 IC50 = 97.18 nM T64969 CNGZ92 127052993 IC50 = 2.92 nM T64969 CBHF87 127052994 IC50 = 62 nM T64969 CS5T2B 127053079 IC50 = 37.81 nM T64969 CIU72D 127264586 IC50 = 5.3 nM T64969 C8ZM1T 129281909 IC50 = 3.6 nM T64969 C2LWZ1 129318964 IC50 > 10000 nM T64969 C0XS4M 129896681 IC50 > 10000 nM T64969 C0FM1R 130196825 IC50 = 1970 nM T64969 CGOQ27 130412632 IC50 = 1.6 nM T64969 CFA3V6 132020316 IC50 = 73.1 nM T64969 CUO0C5 132156633 IC50 > 10000 nM T64969 CV8DP9 132487332 IC50 = 3.23 nM T64969 C0G9TV 132495274 IC50 = 0.12 nM T64969 C51EID 132496692 IC50 < 0.5 nM T64969 C0V2WX 132578497 IC50 = 3.3 nM T64969 CRV07S 132597737 IC50 = 0.3 nM T64969 CL6E4J 132601725 IC50 > 25000 nM T64969 C53OJM 132607333 IC50 = 980.83 nM T64969 CA6TN4 132609257 IC50 = 6.4 nM T64969 CMI3Q0 132819888 IC50 = 690 nM T64969 CERS64 132937256 IC50 > 30000 nM T64969 C46ORZ 132938092 IC50 = 21 nM T64969 C32QRI 132938093 IC50 = 11 nM T64969 CN9SD7 132942957 IC50 = 92.5 nM T64969 CMP2S9 132942958 IC50 = 7.2 nM T64969 CDMF97 134130282 IC50 > 150000 nM T64969 C2H6PW 134130554 IC50 > 150000 nM T64969 CM5T6K 134130825 IC50 = 8 nM T64969 CWF16B 134131331 IC50 > 100000 nM T64969 CLV5I3 134131586 IC50 > 150000 nM T64969 C79SPC 134131685 IC50 = 5200 nM T64969 CC1EB5 134131929 IC50 = 4 nM T64969 CTC7P8 134132114 IC50 = 11 nM T64969 CHW59N 134132187 IC50 = 240 nM T64969 CE1Y8U 134132335 IC50 = 280 nM T64969 CA7J2D 134132574 IC50 = 4.2 nM T64969 C6CYV4 134132651 IC50 > 10000 nM T64969 C3NEU6 134133052 IC50 = 86 nM T64969 CS79UR 134133060 IC50 = 460 nM T64969 C1BTI2 134133235 IC50 = 5.4 nM T64969 CMZG34 134133313 IC50 = 8 nM T64969 C1VOY4 134133329 IC50 = 8 nM T64969 C6IU4F 134133491 IC50 = 500 nM T64969 CZT6O0 134133815 IC50 = 4.6 nM T64969 CI53QU 134133842 IC50 = 64 nM T64969 CG8M5O 134134176 IC50 = 130 nM T64969 CX2WN6 134134364 IC50 = 16 nM T64969 CTZ84R 134134811 IC50 = 4700 nM T64969 C15PJY 134134898 IC50 = 0.4 nM T64969 CH3QN8 134135021 IC50 = 5.6 nM T64969 CPJG85 134135151 IC50 = 601 nM T64969 C3COF8 134135258 IC50 = 4.4 nM T64969 CSZX25 134135323 IC50 = 16 nM T64969 CR5F3L 134135362 IC50 = 668 nM T64969 CDMJ75 134135414 IC50 = 3.6 nM T64969 CV4Q0M 134135529 IC50 = 763 nM T64969 CEQ1M7 134135734 IC50 = 235 nM T64969 CF9NZ6 134135902 IC50 = 118.7 nM T64969 CUL3Q0 134136044 IC50 = 300 nM T64969 C1GVQ7 134136098 IC50 = 175 nM T64969 C3G7TQ 134136245 IC50 = 36 nM T64969 CUP13V 134136269 IC50 = 0.6 nM T64969 CD1O7N 134136322 IC50 = 4649 nM T64969 CZD0J5 134136450 IC50 = 8500 nM T64969 C3LX0Z 134136666 IC50 = 47 nM T64969 C9FZ3A 134136788 IC50 = 587 nM T64969 CL4PT1 134137211 IC50 > 10000 nM T64969 CG92RQ 134137314 IC50 = 593 nM T64969 CYGZ85 134137500 IC50 = 10 nM T64969 CN79XJ 134137614 IC50 = 78 nM T64969 C1U2MV 134137679 IC50 = 460 nM T64969 CJC1E8 134137789 IC50 = 6.4 nM T64969 CK15UI 134137837 IC50 = 502 nM T64969 CJ7C1N 134137974 IC50 = 14 nM T64969 C2L8OB 134138134 IC50 = 510 nM T64969 CC86FV 134138222 IC50 = 136 nM T64969 C3RA6C 134138227 IC50 = 0.27 nM T64969 C5JH9E 134138228 IC50 = 29 nM T64969 CY3U6V 134138310 IC50 = 36 nM T64969 CTY21M 134138472 IC50 = 98.2 nM T64969 CC42DJ 134138534 IC50 = 22 nM T64969 C4QSZ5 134138566 IC50 = 29 nM T64969 CZU97C 134138682 IC50 = 2 nM T64969 C0GT4V 134138751 IC50 = 9 nM T64969 CLG84S 134138800 IC50 = 5.3 nM T64969 C6RGN8 134138812 IC50 = 30 nM T64969 C58FUC 134139047 IC50 = 2 nM T64969 C45HRS 134139393 IC50 = 194 nM T64969 CG91IQ 134139430 IC50 = 79 nM T64969 C5OEI3 134139438 IC50 = 23 nM T64969 C6U5WE 134139490 IC50 = 94 nM T64969 CA7PD8 134139534 IC50 = 857 nM T64969 C3OBC6 134139548 IC50 = 61 nM T64969 C59COE 134139584 IC50 = 1.5 nM T64969 C81QJV 134139647 IC50 = 75 nM T64969 CW69GT 134139694 IC50 = 8 nM T64969 CQE08L 134139702 IC50 = 9 nM T64969 CK7EZ2 134139706 IC50 = 5.8 nM T64969 CO9W1Q 134139995 IC50 = 20 nM T64969 CHL7B1 134140023 IC50 > 1000 nM T64969 CJ9RI1 134140064 IC50 = 51 nM T64969 C8JR1X 134140108 IC50 = 7 nM T64969 C6M9DN 134140179 IC50 = 570 nM T64969 C1QSH4 134140222 IC50 = 1370 nM T64969 CCF0X1 134140501 IC50 = 0.65 nM T64969 C6UJG4 134140680 IC50 = 116 nM T64969 CI2L7Z 134140949 IC50 = 522 nM T64969 C1OB7Z 134141093 IC50 = 100.6 nM T64969 CFAW82 134141290 IC50 = 140 nM T64969 C6HD9W 134141630 IC50 = 53 nM T64969 CM05IQ 134141901 IC50 = 2 nM T64969 CLV6A3 134141947 IC50 = 24 nM T64969 C8KC5F 134142230 IC50 = 898 nM T64969 CS95WZ 134142314 IC50 = 9941 nM T64969 CP38FT 134142454 IC50 > 10000 nM T64969 CC3I0G 134142769 IC50 = 6400 nM T64969 CI92TY 134142809 IC50 = 870 nM T64969 C7TF6I 134142952 IC50 = 4.1 nM T64969 CJT12G 134143005 IC50 = 42 nM T64969 CY9M7L 134143068 IC50 = 747 nM T64969 CSTC29 134143257 IC50 = 509 nM T64969 C4F6VU 134143525 IC50 = 26 nM T64969 C92VFI 134143736 IC50 = 260 nM T64969 CZNJ57 134143863 IC50 = 4.6 nM T64969 CMV45A 134144196 IC50 = 2.7 nM T64969 CWS6V1 134144330 IC50 = 24 nM T64969 C0BJ1U 134144565 IC50 = 9.1 nM T64969 CGD4S5 134144603 IC50 = 28 nM T64969 CH1S3B 134144825 IC50 = 40.6 nM T64969 C38JMR 134145160 IC50 = 531 nM T64969 CO7LU3 134145579 IC50 = 383 nM T64969 CB89WK 134145650 IC50 > 10000 nM T64969 C0TYW7 134145741 IC50 = 388 nM T64969 C1OYR9 134145751 IC50 = 65 nM T64969 CBC06T 134145933 IC50 = 14 nM T64969 CVO98Y 134145943 IC50 > 100 nM T64969 CKZ2I0 134145988 IC50 = 593 nM T64969 CRZ0E5 134146010 IC50 = 8 nM T64969 CZP47U 134146163 IC50 = 160 nM T64969 CTMJ14 134146542 IC50 = 881 nM T64969 CN35SO 134146628 IC50 > 1000 nM T64969 CHJ13S 134146699 IC50 = 19 nM T64969 C0KNV3 134146887 IC50 = 3 nM T64969 CS7CJ4 134146891 IC50 = 212 nM T64969 C3K4ME 134147150 IC50 = 7 nM T64969 C4U8KT 134147234 IC50 = 7 nM T64969 CDF1R9 134147522 IC50 > 10000 nM T64969 CS0WH4 134147608 IC50 = 6.7 nM T64969 C5C9UN 134147625 IC50 = 140 nM T64969 CJ1FQ6 134147869 IC50 = 3 nM T64969 CXS38A 134147887 IC50 = 2 nM T64969 CUKE45 134147919 IC50 > 10000 nM T64969 C4ID3S 134148105 IC50 = 7 nM T64969 CZT40L 134148122 IC50 = 4 nM T64969 CZD10T 134148132 IC50 = 106 nM T64969 CPGL96 134148137 IC50 = 17 nM T64969 CDCJ80 134148182 IC50 > 1000 nM T64969 CN4HT6 134148374 IC50 = 330 nM T64969 CGVC01 134148454 IC50 = 714 nM T64969 CH8A5L 134148508 IC50 = 90 nM T64969 CH5O1F 134148524 IC50 = 15 nM T64969 C5R2PK 134148588 IC50 = 390 nM T64969 C0AWH3 134148660 IC50 = 10 nM T64969 CS0J8U 134148764 IC50 > 1000 nM T64969 CFZI08 134149229 IC50 = 817 nM T64969 C3AS1E 134149331 IC50 = 74 nM T64969 CP14DK 134149339 IC50 = 6.9 nM T64969 CRBI31 134149577 IC50 = 77 nM T64969 CIMW36 134149689 IC50 = 56 nM T64969 CU7FX1 134149906 IC50 = 6.3 nM T64969 C6B4YD 134149918 IC50 = 13 nM T64969 C6Z2JL 134149963 IC50 = 86 nM T64969 CE69LC 134150331 IC50 = 10 nM T64969 CIKN06 134150340 IC50 = 6.9 nM T64969 CQ03OC 134150381 IC50 = 10 nM T64969 CJ56EZ 134150417 IC50 = 1 nM T64969 CM7H0R 134150543 IC50 = 1.9 nM T64969 C1PDA8 134150559 IC50 = 470 nM T64969 CQK40B 134150618 IC50 = 10 nM T64969 C6CFO5 134150713 IC50 = 1 nM T64969 CA4SQ5 134151152 IC50 = 6 nM T64969 C76JIM 134151200 IC50 > 10000 nM T64969 C7CT2Y 134151327 IC50 = 61 nM T64969 CRH2V4 134151618 IC50 = 84 nM T64969 C7NB0Z 134152247 IC50 = 611 nM T64969 CU5T1N 134152381 IC50 > 10000 nM T64969 CG10PO 134152385 IC50 = 77 nM T64969 CI4A1T 134152401 IC50 = 12 nM T64969 CJ9N1A 134152440 IC50 = 14 nM T64969 C76WDH 134152470 IC50 = 44 nM T64969 CWT0Q7 134152512 IC50 > 100 nM T64969 CM62UF 134152586 IC50 = 103.4 nM T64969 C34KQM 134152648 IC50 = 6 nM T64969 C0N6JF 134152887 IC50 = 14 nM T64969 C9ORY0 134152991 IC50 = 21 nM T64969 CW6A7E 134153017 IC50 = 343 nM T64969 C5WV9Z 134153022 IC50 = 22 nM T64969 CLBK62 134153313 IC50 = 65 nM T64969 CLRD90 134153659 IC50 = 27 nM T64969 C1XJ7U 134153922 IC50 = 86 nM T64969 C6JFN5 134153988 IC50 = 72 nM T64969 CR09XE 134154074 IC50 = 88 nM T64969 C8Z3DN 134154342 IC50 = 21 nM T64969 C2Q1XW 134154347 IC50 = 36 nM T64969 CET5R1 134154580 IC50 = 184 nM T64969 C5YX7T 134154596 IC50 = 26 nM T64969 CTG04X 134154708 IC50 = 4 nM T64969 C07RWN 134154721 IC50 = 14 nM T64969 CV5M1T 134154754 IC50 = 5 nM T64969 CI0S4B 134155078 IC50 = 67 nM T64969 C2ISW7 134155088 IC50 = 1 nM T64969 CMH0X4 134155167 IC50 = 519 nM T64969 C48UIX 134155220 IC50 = 9 nM T64969 CVA34W 134155401 IC50 = 2 nM T64969 CR54HK 134155423 IC50 = 17 nM T64969 CJW2N9 134155488 IC50 = 1.1 nM T64969 C9DRQ6 134155700 IC50 = 60 nM T64969 C90IBM 134155874 IC50 = 9300 nM T64969 C6HN5J 134155932 IC50 = 12 nM T64969 CBY2R8 134156011 IC50 = 0.69 nM T64969 CS56YR 134156100 IC50 = 421 nM T64969 C4ZUO0 134156542 IC50 = 93 nM T64969 C2QN7B 134156570 IC50 = 2933 nM T64969 CKL8X3 134156658 IC50 = 45 nM T64969 CF7KA3 134156808 IC50 = 109 nM T64969 CQD93J 134156816 IC50 = 21 nM T64969 C3HCT6 134156845 IC50 = 25 nM T64969 CI4W7T 134156856 IC50 = 11.6 nM T64969 CH1GS2 134157091 IC50 = 6.5 nM T64969 COVM37 134157236 IC50 > 10000 nM T64969 CF85NI 134157315 IC50 = 205 nM T64969 CEHV70 134157345 IC50 = 19 nM T64969 CG36DX 134157614 IC50 = 127 nM T64969 C2AN7T 134611886 IC50 > 100000 nM T64969 CZ8W6R 134612705 IC50 > 1000 nM T64969 CYL5V1 134694986 IC50 > 30000 nM T64969 CG15PY 134812846 IC50 > 50000 nM T64969 CN3Y9J 134817166 IC50 = 1.1 nM T64969 COK96J 134827795 IC50 = 17 nM T64969 CIZ39M 134827836 IC50 > 100000 nM T64969 CJ04NP 134827837 IC50 = 140 nM T64969 C54FXD 134957362 IC50 > 10000 nM T64969 CUL3M1 134959408 Ki = 0.1 nM T64969 C82ENU 135128874 Ki = 105 nM T64969 C0NCM1 135236452 IC50 = 6.5 nM T64969 C7EMI6 135236457 IC50 = 210 nM T64969 CWBO79 135236483 IC50 = 219 nM T64969 CH3ZB7 135236498 IC50 = 5.8 nM T64969 CXDY80 135236566 IC50 = 9 nM T64969 C5SEK3 135236586 IC50 = 199 nM T64969 CIOD87 135236597 IC50 = 413 nM T64969 C45LFT 135236603 IC50 = 300 nM T64969 CR9TH8 135236627 IC50 > 10000 nM T64969 C3J5LM 135236635 IC50 = 20 nM T64969 CB6EG0 135236676 IC50 = 8630 nM T64969 CL93ZY 135236756 IC50 = 420 nM T64969 C0DV1Q 135236809 IC50 = 36 nM T64969 CS4BM3 135236903 IC50 = 10.9 nM T64969 CGJ07D 135236905 IC50 = 48 nM T64969 CNC56O 135251923 IC50 = 26.8 nM T64969 C2PH4R 135251924 IC50 = 494 nM T64969 CO43PJ 135251926 IC50 = 730 nM T64969 C4IO8Z 135313938 Ki = 0.03 nM T64969 C6IYG1 135314117 IC50 < 1 nM T64969 CCM74D 135369110 IC50 = 46.5 nM T64969 C4PN7O 135400972 IC50 = 50000 nM T64969 CVJK60 135402835 IC50 = 6 nM T64969 CPE8O5 135402837 IC50 = 588 nM T64969 CO3H4I 135402838 IC50 = 0.17 nM T64969 CK67RJ 135402839 IC50 = 4.7 nM T64969 C05WPI 135402840 IC50 = 1.24 nM T64969 C38ASJ 135402848 IC50 = 346.74 nM T64969 CLFE42 135402849 IC50 = 1.6 nM T64969 CJ1I5M 135402981 IC50 > 1000 nM T64969 CH97JB 135402982 IC50 > 1000 nM T64969 C26GSU 135402983 IC50 > 1000 nM T64969 CK8EJ6 135402984 IC50 > 1000 nM T64969 C1Q9SE 135407125 IC50 = 130000 nM T64969 CAZ5X6 135407149 IC50 = 60000 nM T64969 CR3XN0 135408977 IC50 = 3100 nM T64969 C7LI1N 135408978 IC50 = 1400 nM T64969 CQ54JK 135410197 IC50 = 71700 nM T64969 CQ4RD2 135410274 IC50 > 10000 nM T64969 CUI1B3 135417010 IC50 = 7700 nM T64969 CK9D4A 135428921 EC50 = 33000 nM T64969 C85SLV 135430346 IC50 = 20 ug.mL-1 T64969 COI9Y2 135431544 IC50 = 5300 nM T64969 CU60YC 135431661 IC50 > 30000 nM T64969 C5FO9E 135433976 IC50 = 30000 nM T64969 C4VH8I 135438239 IC50 = 5600 nM T64969 C16XLU 135454992 IC50 > 10000 nM T64969 CIP6W1 135457450 IC50 = 10000 nM T64969 CIJ9Q2 135461535 IC50 = 3920 nM T64969 C3WK8O 135464283 IC50 = 61000 nM T64969 CX35PB 135468746 IC50 > 100000 nM T64969 C01NXG 135469322 IC50 = 58000 nM T64969 CMU4G6 135474309 IC50 = 27000 nM T64969 CWPK94 135478626 IC50 = 1400 nM T64969 CRTS92 135484881 IC50 > 100000 nM T64969 CGXS54 135485502 IC50 = 75000 nM T64969 CMOR61 135492395 IC50 > 10000 nM T64969 CKF6R5 135492549 IC50 >> 2000 nM T64969 CJB83H 135494293 IC50 = 6 ug.mL-1 T64969 CCOL98 135499946 IC50 = 100000 nM T64969 C64EMD 135500075 IC50 > 10000 nM T64969 CH91IT 135503554 IC50 > 10000 nM T64969 CP0R1O 135503606 IC50 > 100000 nM T64969 CVZ08D 135509841 IC50 > 10000 nM T64969 CYQ5M6 135511836 IC50 = 300000 nM T64969 CGI1H3 135516745 IC50 = 20000 nM T64969 C5TW9S 135517293 IC50 >> 10000 nM T64969 CG1WR0 135518082 IC50 = 130000 nM T64969 CJI0G1 135520135 IC50 > 10000 nM T64969 CLK9D1 135523696 IC50 = 75000 nM T64969 CTJ48K 135524085 IC50 = 3300 nM T64969 CUT1W7 135524168 IC50 > 10000 nM T64969 CRT3X6 135524445 IC50 = 2100 nM T64969 CIA18F 135525349 IC50 = 5000 nM T64969 CIM0Q6 135526986 IC50 > 20000 nM T64969 C3XK7R 135531249 IC50 = 8.5 ug.mL-1 T64969 C2MAC7 135536640 IC50 > 100000 nM T64969 COXH29 135543616 IC50 >> 20000 nM T64969 CM72XH 135546247 IC50 = 20 ug.mL-1 T64969 C0J3BN 135678111 IC50 > 50000 nM T64969 CU29YK 135750268 IC50 = 922 nM T64969 CX4ZB3 135863110 IC50 > 10000 nM T64969 CM3UC9 135883136 IC50 = 370 nM T64969 C8LN7E 135883350 IC50 > 100000 nM T64969 CUV73C 135883354 IC50 > 100000 nM T64969 CIPA79 135937899 IC50 = 2200 nM T64969 C12UDA 135947972 IC50 = 1040 nM T64969 CN42ZS 135947973 IC50 = 954 nM T64969 CF8AO3 135947974 IC50 = 6900 nM T64969 CW08GJ 135947976 IC50 = 7400 nM T64969 CJN7E2 135947978 IC50 = 908 nM T64969 CFKH34 135947979 IC50 = 88 nM T64969 C2PAV1 135971426 IC50 = 3300 nM T64969 C9W6BT 136002660 IC50 = 10900 nM T64969 CD9CT6 136002661 IC50 = 989 nM T64969 C4T9KZ 136002662 IC50 = 726 nM T64969 CHA4N2 136013680 IC50 > 10 nM T64969 CLN6Y8 136026516 IC50 > 100000 nM T64969 CQ0KD1 136036218 IC50 = 1.585 nM T64969 CGP0K5 136036219 IC50 = 0.4169 nM T64969 C2ZX7P 136036220 IC50 = 0.912 nM T64969 C4HNF6 136036221 IC50 = 5.754 nM T64969 C67UGS 136036222 IC50 = 3.631 nM T64969 CLZ9Q1 136036223 IC50 = 0.4786 nM T64969 C3N4KU 136036228 IC50 = 0.7244 nM T64969 C5AY0R 136036229 IC50 = 0.7762 nM T64969 CH0AO1 136042228 IC50 = 34250 nM T64969 CJ7U4C 136053657 IC50 > 100000 nM T64969 CZP3W5 136066077 IC50 = 28.5 nM T64969 C8D0YV 136066078 IC50 = 3.16 nM T64969 C4LGS1 136066079 IC50 = 65.5 nM T64969 CCAM43 136066080 IC50 = 4.45 nM T64969 CIG6B4 136066100 IC50 = 16.9 nM T64969 CBH08O 136066101 IC50 = 23.8 nM T64969 CG1R7B 136087060 IC50 > 10000 nM T64969 CGP69Y 136130281 IC50 = 501187.23 nM T64969 CH64ID 136175114 IC50 > 10000 nM T64969 CDT7E4 136211077 IC50 > 1000 nM T64969 C9RE8D 136215817 IC50 > 100000 nM T64969 C1YUD0 136219394 IC50 > 10 nM T64969 C5QAT2 136236302 IC50 = 24.1 nM T64969 CIU8W3 136254389 IC50 > 10 nM T64969 CRK8E5 136391507 IC50 = 0.48 nM T64969 CR69AU 136928128 IC50 = 0.63 nM T64969 C03VDE 136928142 IC50 = 141 nM T64969 CTAS87 136983688 IC50 = 2.1 nM T64969 C8M2DL 136983691 IC50 = 169 nM T64969 CMOH82 136983718 IC50 = 0.18 nM T64969 C1JSX0 136983721 IC50 = 0.46 nM T64969 CRE05Z 136983730 IC50 = 3.1 nM T64969 CMP62O 136983732 IC50 = 0.3 nM T64969 CB26DO 136983736 IC50 = 0.66 nM T64969 C9J5KZ 136983740 IC50 = 0.34 nM T64969 CN7W2C 136983741 IC50 = 1.2 nM T64969 CPM64E 136983746 IC50 = 0.79 nM T64969 CM2IO7 136983748 IC50 < 0.25 nM T64969 C60HNV 136983761 IC50 = 3.2 nM T64969 C4EKW0 136983767 IC50 = 21 nM T64969 C69LHV 137175062 Ki = 58 nM T64969 C41AYR 137175217 Ki = 88 nM T64969 C83WAK 137189946 IC50 = 3600 nM T64969 C0LR2H 137189948 IC50 > 20000 nM T64969 C8KW0I 137189951 IC50 = 3450 nM T64969 COX23B 137189952 IC50 = 4390 nM T64969 CSGM03 137210056 IC50 > 10000 nM T64969 CXT8B9 137287443 IC50 = 51 nM T64969 C2SY8T 137302575 IC50 = 3 nM T64969 CUL6Z7 137319850 IC50 < 1 nM T64969 C3Z4AT 137321159 IC50 > 10000 nM T64969 CE75QD 137321162 IC50 = 520 nM T64969 CM4TU2 137321167 IC50 = 30 nM T64969 CWH6I2 137348469 IC50 = 2.5 nM T64969 CF2B4A 137348470 IC50 = 1 nM T64969 CKC2Q5 137348686 IC50 = 649 nM T64969 C6A8BE 137349495 IC50 = 690 nM T64969 C9OQ2L 137436777 IC50 = 168.8 nM T64969 CPYC42 137436898 IC50 > 1000 nM T64969 CZL7X1 137436936 IC50 = 65.1 nM T64969 C1KSZ6 137475463 IC50 = 5882 nM T64969 C2FT1L 137475480 IC50 = 6863 nM T64969 C13DTZ 137628688 IC50 = 5.8 nM T64969 C6V3UK 137631426 IC50 = 11.3 nM T64969 C58XRH 137631553 IC50 = 23.99 nM T64969 CZE86J 137631564 IC50 = 183 nM T64969 CMP5H4 137631852 IC50 > 10000 nM T64969 C0CE4R 137631936 IC50 = 2 nM T64969 C81MHK 137631947 IC50 = 48.9 nM T64969 C25ERN 137631967 IC50 = 4.2 nM T64969 CK9TO3 137632059 IC50 = 10.2 nM T64969 CH9WK1 137632228 IC50 > 10000 nM T64969 CW2I0X 137632429 IC50 = 28.9 nM T64969 C6HYQ4 137632485 IC50 = 373.7 nM T64969 CNO0W6 137632514 IC50 = 46 nM T64969 C6BWP9 137632530 IC50 = 297 nM T64969 C8YXN5 137632579 IC50 = 10.2 nM T64969 C9Y4UW 137632652 IC50 = 15.4 nM T64969 CX4BG3 137632686 IC50 = 257 nM T64969 C1IRD9 137632976 IC50 = 600 nM T64969 COW53U 137633148 IC50 = 60.1 nM T64969 C8J5YE 137633149 IC50 = 60953.69 nM T64969 C52PDU 137633245 IC50 = 100000 nM T64969 CAW72M 137633292 IC50 = 3400 nM T64969 CWP23Z 137633367 IC50 = 5700 nM T64969 C6W9VB 137633473 IC50 < 1 nM T64969 CKD94A 137633488 IC50 = 65400 nM T64969 CFUY16 137633842 IC50 = 4300 nM T64969 C41TLP 137634049 IC50 = 188.2 nM T64969 CNX0F9 137634126 IC50 = 360 nM T64969 CHC70D 137634143 IC50 = 725.3 nM T64969 C3Z5UO 137634208 IC50 = 8470 nM T64969 CI1E8V 137634241 IC50 > 10000 nM T64969 CE9G6I 137634299 IC50 = 120 nM T64969 CD64EL 137634342 IC50 = 25.3 nM T64969 C58JAF 137634409 IC50 = 549.6 nM T64969 CFP2A7 137634412 IC50 = 100000 nM T64969 CM3JB8 137634462 IC50 > 150 nM T64969 CP0J4V 137634715 IC50 = 10 nM T64969 C42PMG 137634834 IC50 = 52.8 nM T64969 C2DT0F 137634837 IC50 = 413 nM T64969 C9MJB3 137635188 IC50 = 17.6 nM T64969 CKH35C 137635255 Ki = 3680 nM T64969 C18FSE 137635348 IC50 = 28.7 nM T64969 CICR67 137635590 IC50 = 14.2 nM T64969 C42CPG 137635606 IC50 < 1 nM T64969 CS23KQ 137635618 IC50 = 20000 nM T64969 CY4M7O 137635632 Ki = 640 nM T64969 CI8T3V 137635635 IC50 = 1120 nM T64969 C5JD9N 137635898 IC50 = 2.3 nM T64969 C61KRW 137636025 IC50 = 5900 nM T64969 CW03UM 137636140 IC50 = 10 nM T64969 C1UM2S 137636157 IC50 > 150 nM T64969 CL4US7 137636248 IC50 > 150 nM T64969 C6LB3K 137636403 IC50 = 100000 nM T64969 CY6S7J 137636429 IC50 = 26.9 nM T64969 CVD9E7 137636479 IC50 = 60 nM T64969 C1EXD3 137636509 IC50 = 67.9 nM T64969 CB89IY 137636527 IC50 > 100000 nM T64969 CPF75D 137636602 IC50 = 55.5 nM T64969 C2IOU5 137636607 IC50 = 26 nM T64969 CXLM63 137636621 IC50 < 0.3 nM T64969 C2FA3S 137636658 IC50 = 4050 nM T64969 CT17QN 137636787 IC50 = 2.3 nM T64969 C8BDC7 137636863 IC50 = 7 nM T64969 C9K5AS 137637051 IC50 = 28 nM T64969 C06JRX 137637094 IC50 = 4.7 nM T64969 CXJ3Q0 137637114 IC50 = 6.13 nM T64969 CRD5K6 137637150 IC50 = 20 nM T64969 CB9MO6 137637177 IC50 = 1.8 nM T64969 C5LU2S 137637274 Ki = 80 nM T64969 CSC2Q3 137637327 IC50 = 12 nM T64969 C0YD2I 137637558 IC50 = 467 nM T64969 CJ86NK 137637579 IC50 = 55 nM T64969 C63SHA 137637655 IC50 = 56 nM T64969 CT7BW5 137637707 IC50 < 1 nM T64969 C36UDX 137637748 IC50 = 25 nM T64969 CRXH80 137637913 IC50 = 1 nM T64969 CIPT52 137638089 IC50 = 0.5 nM T64969 CGNL27 137638186 IC50 = 1.9 nM T64969 CSU32D 137638440 IC50 = 7.8 nM T64969 CD7ZQ9 137638445 IC50 = 120 nM T64969 CU24QC 137638448 IC50 = 33.6 nM T64969 C4NBP2 137638482 IC50 = 11.2 nM T64969 CI45NR 137638579 IC50 = 133.1 nM T64969 CDHR26 137638664 IC50 = 1300 nM T64969 CSC8I9 137638715 IC50 = 120 nM T64969 CG09DY 137638779 IC50 = 27.4 nM T64969 CIAL90 137638797 IC50 < 1 nM T64969 C8G0XY 137638840 IC50 = 97 nM T64969 C3FU9S 137638860 IC50 = 436.3 nM T64969 CS8I4L 137639015 IC50 = 595.2 nM T64969 CB9K0T 137639063 IC50 > 150 nM T64969 CLWZ62 137639100 IC50 = 1.6 nM T64969 CLM2E7 137639118 IC50 < 0.3 nM T64969 CDG3W9 137639160 Ki = 5950 nM T64969 C1CJL8 137639161 IC50 = 302 nM T64969 CTQ2Y9 137639273 IC50 > 150 nM T64969 CM12TX 137639299 IC50 = 36.8 nM T64969 CZ4JS5 137639379 Ki = 370 nM T64969 CE75PY 137639383 IC50 = 3.3 nM T64969 CBM75H 137639408 IC50 = 35.8 nM T64969 C39GHY 137639513 Ki = 0.38 nM T64969 C3UBE2 137639638 IC50 = 47.1 nM T64969 CE96AL 137639657 IC50 = 3.2 nM T64969 CEWX78 137639774 IC50 = 34320 nM T64969 C9QS8P 137639893 IC50 > 150 nM T64969 C0GI7M 137639998 Ki = 290 nM T64969 CZ3RG6 137640107 IC50 = 28.3 nM T64969 CUQ32R 137640370 IC50 = 1.9 nM T64969 CP4WE6 137640788 IC50 = 4.53 nM T64969 CEPC29 137640799 IC50 = 220 nM T64969 C3PBM5 137640804 IC50 = 20 nM T64969 CZA04C 137640806 IC50 = 2000 nM T64969 C6LE5P 137640904 Ki = 610 nM T64969 C45TDX 137641093 IC50 = 287 nM T64969 CI9A6R 137641259 IC50 = 26.5 nM T64969 CF0B2T 137641286 IC50 = 137 nM T64969 C7TG3J 137641313 IC50 > 19952.62 nM T64969 CM0ID8 137641315 IC50 = 100000 nM T64969 C2S5HW 137641579 IC50 = 200 nM T64969 CADV57 137641678 IC50 = 22 nM T64969 CC7NA3 137641695 IC50 = 7.6 nM T64969 C4S0NY 137641776 IC50 = 20 nM T64969 CDF05B 137641797 IC50 = 1600 nM T64969 CI48MT 137641870 IC50 = 15.69 nM T64969 CO7T1M 137642099 IC50 = 35.4 nM T64969 CA26QR 137642204 IC50 = 217 nM T64969 CE78MV 137642234 IC50 = 10 nM T64969 CFP6S7 137642384 IC50 = 132.1 nM T64969 C0M2DV 137642413 IC50 = 2900 nM T64969 CHSF21 137642481 IC50 = 6 nM T64969 CYIM43 137642492 IC50 = 46300 nM T64969 CG0P7F 137642583 IC50 < 0.3 nM T64969 C1BEM9 137642718 IC50 = 0.8 nM T64969 CR7DU4 137642765 Ki = 910 nM T64969 C04WMX 137642837 IC50 < 1 nM T64969 C86ZQY 137642882 IC50 = 46.8 nM T64969 CU6V4B 137642950 IC50 = 86200 nM T64969 CU8YX6 137643005 IC50 = 167300 nM T64969 CEX71A 137643024 IC50 = 889 nM T64969 C3VE1J 137643259 IC50 = 19.3 nM T64969 CC24DF 137643392 IC50 = 838.5 nM T64969 C1TN5U 137643437 IC50 = 127.8 nM T64969 CO2WA8 137643441 IC50 = 1.1 nM T64969 C5NB8J 137643535 IC50 = 100000 nM T64969 CSJ4F0 137643599 IC50 = 295.7 nM T64969 C9KC1X 137643767 IC50 = 2626 nM T64969 CZN72T 137644087 IC50 = 222.5 nM T64969 CRQL24 137644097 IC50 = 100000 nM T64969 CNK3C1 137644195 IC50 = 24.4 nM T64969 CGV72K 137644347 IC50 > 150 nM T64969 CV8G5N 137644357 IC50 < 1 nM T64969 CJ6I3O 137644466 IC50 = 1.1 nM T64969 CVP54C 137644489 IC50 = 6.2 nM T64969 CQ08RW 137644617 IC50 = 365 nM T64969 CMEL14 137644727 Ki = 270 nM T64969 CD29JK 137644944 IC50 = 145 nM T64969 C0CSA2 137645004 IC50 = 4.9 nM T64969 COQ1G5 137645019 IC50 = 1.79 nM T64969 CMA01W 137645075 IC50 = 22.2 nM T64969 CS03JL 137645107 IC50 = 60 nM T64969 C15SPX 137645121 IC50 = 100000 nM T64969 CZDI94 137645280 IC50 = 1900 nM T64969 CCG29K 137645358 IC50 = 3210 nM T64969 CKP7N9 137645385 Ki = 1260 nM T64969 C27ISW 137645443 IC50 = 60.7 nM T64969 C37UPA 137645513 IC50 = 40 nM T64969 C9RY1I 137645557 IC50 = 16 nM T64969 CW5N0Q 137645598 IC50 = 40 nM T64969 C7Q0KP 137645669 IC50 = 373 nM T64969 CJ94TQ 137645832 IC50 = 7230 nM T64969 CQJ45H 137645835 IC50 = 26.6 nM T64969 CT4JK0 137645956 IC50 = 14.5 nM T64969 C03VKP 137646019 IC50 < 1 nM T64969 CFVP34 137646278 Ki = 110 nM T64969 CHL6W7 137646293 IC50 = 36.9 nM T64969 CX9QM0 137646296 Ki = 900 nM T64969 CN2J6Z 137646310 IC50 = 365 nM T64969 C7K6XE 137646529 IC50 > 10000 nM T64969 CDK1X9 137646546 IC50 = 3400 nM T64969 CSEV89 137646548 IC50 = 45 nM T64969 CS6J0V 137646549 IC50 = 98 nM T64969 CB45FK 137646625 IC50 = 15 nM T64969 C1MJ2B 137646681 IC50 = 2.6 nM T64969 C39ECO 137646754 IC50 = 33189.45 nM T64969 CE2GS1 137646967 IC50 = 117.5 nM T64969 CNR6Y9 137647154 IC50 = 427.7 nM T64969 C84XPS 137647374 IC50 = 63.6 nM T64969 CRI7W4 137647547 IC50 = 25.5 nM T64969 C1MO6F 137647858 IC50 = 153 nM T64969 CV34AT 137647876 IC50 = 4700 nM T64969 CB4G7L 137648004 IC50 = 979.49 nM T64969 CHKS97 137648071 Ki = 90 nM T64969 CB02WE 137648106 IC50 = 87 nM T64969 CHYD27 137648384 IC50 = 10.9 nM T64969 C4Q5FE 137648385 IC50 < 0.5 nM T64969 CZO42N 137648629 IC50 > 100000 nM T64969 CDWM98 137648631 IC50 = 209 nM T64969 CNZV16 137648828 IC50 = 4.5 nM T64969 CA1H0Y 137649110 IC50 = 18.7 nM T64969 CPY41L 137649188 IC50 = 102 nM T64969 CQ53DI 137649227 IC50 = 210 nM T64969 CQ2D4K 137649247 IC50 = 8.9 nM T64969 CRL38H 137649329 IC50 = 146.3 nM T64969 CWAP61 137649410 IC50 = 24 nM T64969 CZ5DB2 137649455 IC50 = 9.5 nM T64969 C3XQ4T 137649572 IC50 = 20 nM T64969 C68MVW 137649573 IC50 = 148 nM T64969 CTBG10 137649803 IC50 = 208.4 nM T64969 CG3D9R 137649880 IC50 = 6.7 nM T64969 CR5JN8 137649915 IC50 = 462 nM T64969 CN3I0J 137650029 IC50 = 130 nM T64969 C6JIK5 137650097 IC50 < 1 nM T64969 CZ5VL9 137650197 IC50 = 100000 nM T64969 CH2R1F 137650251 IC50 = 780 nM T64969 C3UBN8 137650330 IC50 = 3700 nM T64969 CR27SL 137650383 IC50 = 39700 nM T64969 CQ4R1I 137650454 IC50 = 286 nM T64969 CI1U0H 137650532 IC50 = 9.2 nM T64969 C1A6ZV 137650580 IC50 = 218 nM T64969 CX12DJ 137650597 IC50 = 7.2 nM T64969 C4N2VA 137650617 IC50 = 144 nM T64969 C12JHN 137650629 IC50 = 12.1 nM T64969 CS0D7H 137650797 IC50 = 97 nM T64969 CV7WE6 137651016 IC50 = 258 nM T64969 CO6DY4 137651084 IC50 = 2500 nM T64969 C9CZ5R 137651233 IC50 = 22 nM T64969 CM2WA6 137651258 IC50 = 421 nM T64969 C5ZEI9 137651283 IC50 > 150 nM T64969 CX9BD8 137651363 IC50 = 3100 nM T64969 C1DK0P 137651391 IC50 = 8.1 nM T64969 C0IY3L 137651740 IC50 < 1 nM T64969 CUN78O 137651765 IC50 = 5 nM T64969 CBP7D8 137651768 IC50 = 1300 nM T64969 CR0QK4 137651864 IC50 = 15.8 nM T64969 C0GB7L 137651865 IC50 = 1300 nM T64969 CU1WH2 137651878 IC50 = 5.6 nM T64969 C3X0VR 137652014 IC50 = 73500 nM T64969 C2QMD3 137652087 IC50 = 55 nM T64969 C28VPE 137652194 IC50 = 10.71 nM T64969 C6PQ3M 137652198 IC50 = 12 nM T64969 CQUY83 137652218 IC50 = 8300 nM T64969 CO41DK 137652335 IC50 = 673 nM T64969 C7SB9W 137652377 IC50 = 20.6 nM T64969 CJ6S9T 137652622 IC50 = 8.5 nM T64969 C1E0GD 137652646 IC50 = 8.1 nM T64969 CX2L6R 137652830 IC50 = 13 nM T64969 C7Z3OK 137652842 IC50 = 2400 nM T64969 CIK69O 137652848 IC50 = 1.6 nM T64969 CDJ1E5 137652860 IC50 = 1100 nM T64969 C28QUP 137652864 IC50 = 642.7 nM T64969 CW39CF 137652891 IC50 = 57 nM T64969 C3LAD6 137652990 IC50 = 1021 nM T64969 CNB10S 137653041 IC50 = 4900 nM T64969 C9BF1E 137653143 IC50 = 25000 nM T64969 C6RWG4 137653308 IC50 = 4500 nM T64969 CMS31R 137653327 IC50 = 32.35 nM T64969 CZLB29 137653418 IC50 = 100000 nM T64969 C5LV3R 137653430 IC50 = 11 nM T64969 CVF8B2 137653486 IC50 = 9.1 nM T64969 CWFI42 137653795 IC50 = 69984.2 nM T64969 CX3JS6 137653952 IC50 = 278.2 nM T64969 CRSC07 137654213 IC50 = 55.5 nM T64969 CDIG10 137654476 IC50 = 91.8 nM T64969 CHL6R9 137654533 IC50 < 1 nM T64969 C7UEM1 137654543 IC50 = 50000 nM T64969 CUP85I 137654607 IC50 = 518 nM T64969 CST9Z6 137654612 IC50 = 1.2 nM T64969 CZ1D3X 137654743 IC50 > 150 nM T64969 CPMI90 137654861 IC50 = 11 nM T64969 C5CH2P 137654954 IC50 = 216.1 nM T64969 CQGX68 137655106 IC50 = 11.4 nM T64969 CHR5Y4 137655134 IC50 = 29.4 nM T64969 CRN09J 137655337 IC50 = 76 nM T64969 CCXH57 137655416 Ki = 640 nM T64969 C9JT1N 137655519 IC50 = 20800 nM T64969 CO03SP 137655672 IC50 = 32.1 nM T64969 CJHR85 137655678 IC50 = 6900 nM T64969 C5OEN8 137655763 IC50 > 150 nM T64969 CF4BR6 137655863 IC50 = 715 nM T64969 C56LGP 137655890 IC50 = 83.82 nM T64969 CP0EK1 137656130 IC50 > 150 nM T64969 CJ1AL4 137656216 IC50 = 362 nM T64969 C4OL7J 137656236 Ki = 4030 nM T64969 CF65SR 137656304 IC50 = 112.4 nM T64969 CBUK30 137656424 IC50 = 45081.67 nM T64969 CM1X2Z 137656744 IC50 = 5000 nM T64969 COZA85 137656751 IC50 = 80.91 nM T64969 CIP0S1 137656884 IC50 = 10 nM T64969 C02CKX 137656919 IC50 = 888.2 nM T64969 CGK74V 137657167 IC50 = 4.87 nM T64969 CEX13S 137657186 IC50 = 8.9 nM T64969 CKVO51 137657233 IC50 = 4.9 nM T64969 CE2F4M 137657262 IC50 = 383 nM T64969 C4U6BC 137657356 IC50 = 2500 nM T64969 C4L3EC 137657481 IC50 = 0.07 nM T64969 CE3KR1 137657520 IC50 > 150 nM T64969 CWE31H 137657545 IC50 = 417 nM T64969 C2W5XI 137657580 IC50 = 24.9 nM T64969 CV5H3Z 137657932 IC50 = 3.1 nM T64969 CZP9J1 137658032 IC50 = 224.5 nM T64969 C2MCK3 137658120 IC50 = 22 nM T64969 CS14VU 137658122 IC50 = 1200 nM T64969 C64HKO 137658202 IC50 = 23700 nM T64969 CGP0F8 137658204 IC50 < 1 nM T64969 CNM0R5 137658207 IC50 = 0.6 nM T64969 CPV1S9 137658287 IC50 > 1000 nM T64969 CCOQ25 137658337 IC50 = 6.8 nM T64969 CW59EN 137658341 IC50 = 27 nM T64969 C1W3SU 137658355 IC50 = 6.8 nM T64969 CO41NV 137658479 IC50 > 100000 nM T64969 C0T6DR 137658736 IC50 = 19.5 nM T64969 C7IVT9 137658762 IC50 = 167.1 nM T64969 CW89GI 137658864 IC50 < 1 nM T64969 CPD68B 137658974 IC50 > 150 nM T64969 CH5JU3 137658981 IC50 = 23.6 nM T64969 CV2L4Q 137659016 IC50 < 1 nM T64969 C7PL9R 137659061 IC50 = 55.5 nM T64969 CR91LE 137659218 IC50 = 5.7 nM T64969 C2GN1V 137659253 IC50 = 80 nM T64969 C0DC5L 137659278 Ki = 520 nM T64969 CE93JS 137659304 IC50 = 10 nM T64969 CJF6G7 137659313 IC50 = 1100 nM T64969 CC54PL 137659460 IC50 = 17.7 nM T64969 CS61AX 137659496 Ki = 5670 nM T64969 C4HZM7 137659498 IC50 > 150 nM T64969 CJ4YM8 137659634 IC50 = 3.4 nM T64969 C8NZ9V 137659669 IC50 = 75 nM T64969 C73CXG 137659722 IC50 = 15.7 nM T64969 CKL97P 137659725 IC50 = 23.4 nM T64969 CT94YA 137659769 IC50 = 32.1 nM T64969 CS43UI 137659891 IC50 = 15.8 nM T64969 CX2PB5 137660250 IC50 > 150 nM T64969 CBTU32 137660306 IC50 = 360 nM T64969 C46WON 137660327 IC50 > 1000 nM T64969 CLIB19 137660335 IC50 = 33.2 nM T64969 C07JTH 137660356 Ki = 1870 nM T64969 CF41AQ 137660592 IC50 = 4.9 nM T64969 CR4N5S 137660661 IC50 = 1.5 nM T64969 CTZ05I 137660747 IC50 = 11.42 nM T64969 C98GQX 137660836 IC50 = 8.7 nM T64969 C0YZP2 137660958 IC50 < 1 nM T64969 CCO5E1 137660978 IC50 = 10 nM T64969 C89EDU 137661037 IC50 = 6100 nM T64969 C9T8DS 137661049 IC50 = 22 nM T64969 CJ52DB 137661068 IC50 < 1 nM T64969 C1L7BC 137661158 IC50 = 1.9 nM T64969 CKY35O 137661181 Ki = 120 nM T64969 C7PQ6B 137661273 IC50 > 150 nM T64969 CMSH35 137661302 IC50 = 216 nM T64969 CSOE96 137661336 IC50 = 71.6 nM T64969 CM0N3T 137661420 IC50 = 2.6 nM T64969 C2EJB9 137661577 IC50 = 377 nM T64969 CYVS73 137661698 IC50 = 13 nM T64969 CB72MA 137661754 IC50 = 45000 nM T64969 C25FCZ 137661759 IC50 = 33 nM T64969 CT43IF 137661858 IC50 = 1.1 nM T64969 C0Y4XD 137662183 IC50 = 3900 nM T64969 CUY09E 137662185 IC50 = 626 nM T64969 C6CZA9 137662310 IC50 = 700 nM T64969 CM3UF7 137700779 IC50 > 10000 nM T64969 CT1D9K 138454747 IC50 > 1000000 nM T64969 C5LQU9 138479230 IC50 = 384.8 nM T64969 CSRI06 138547901 IC50 > 1000 nM T64969 CUXO19 138617501 IC50 > 1000 nM T64969 C9NYR2 138911325 IC50 = 27.5 nM T64969 CRWA29 139030520 IC50 > 2000 nM T64969 CJI5X1 139447554 IC50 = 12 nM T64969 CDQS68 139447649 IC50 = 519 nM T64969 CSDG73 139447864 IC50 = 353 nM T64969 CZ85HW 139593668 IC50 = 2100 nM T64969 CNI84L 139593669 IC50 = 267 nM T64969 COB9P2 141456067 IC50 > 10000 nM T64969 CWKN18 141489617 IC50 = 7.7 nM T64969 CZ6OQ4 141489621 IC50 = 33.1 nM T64969 C2V3CZ 141489622 IC50 = 142.7 nM T64969 CA6ZE3 141489625 IC50 = 202.3 nM T64969 CTG0M3 141489626 IC50 = 838.5 nM T64969 C42QLX 141489627 IC50 = 38.5 nM T64969 CH74WV 141489632 IC50 > 1000 nM T64969 C8YS7B 141489636 IC50 = 4.1 nM T64969 CZB56Q 141489640 IC50 = 4.1 nM T64969 C9X3BQ 141494014 IC50 = 53.2 nM T64969 CUG0M7 141494019 IC50 = 9.9 nM T64969 CUFX86 141494026 IC50 = 1.5 nM T64969 C4YTS8 141494027 IC50 = 12 nM T64969 CP6ZN9 141494035 IC50 = 1.6 nM T64969 C27MYX 141494043 IC50 = 85 nM T64969 CMND29 141494046 IC50 = 3.9 nM T64969 CT1EH2 141494048 IC50 = 6.5 nM T64969 CHO81S 141494057 IC50 = 3.3 nM T64969 C3SI7W 141494065 IC50 = 2.7 nM T64969 CEVI18 141494066 IC50 = 28.8 nM T64969 CP19EN 141509386 IC50 = 4 nM T64969 CCXT19 141510925 IC50 = 892 nM T64969 C9ED8K 141510928 IC50 = 556 nM T64969 C7TW9O 141510929 IC50 = 114 nM T64969 COLJ50 141510933 IC50 = 104 nM T64969 CI5KY6 141510937 IC50 = 805 nM T64969 CP20DC 141515864 IC50 = 7 nM T64969 CU17OE 141515867 IC50 = 20.7 nM T64969 C34CKN 141523354 IC50 > 10000 nM T64969 CTR7D4 141535114 IC50 = 42.3 nM T64969 CF1R6Z 141725864 IC50 = 7.8 nM T64969 CK35HM 141726486 IC50 = 3.62 nM T64969 C1QB4I 141740774 IC50 = 985 nM T64969 C9T0WU 141740777 IC50 = 37 nM T64969 C4DY2A 141740778 IC50 = 7.5 nM T64969 CMA73H 141740779 IC50 = 1621 nM T64969 COSZ17 141740780 IC50 = 201 nM T64969 CFV8J1 141740781 IC50 = 892 nM T64969 CKIY74 141740782 IC50 > 2000 nM T64969 CEWT18 141740783 IC50 = 977 nM T64969 C7PGK2 141740785 IC50 = 923 nM T64969 CF9N8G 141740786 IC50 = 684 nM T64969 C9XKQ7 141740787 IC50 > 2000 nM T64969 C7M4FY 141740788 IC50 = 1689 nM T64969 C67AUS 141740789 IC50 = 360 nM T64969 CNA8J2 141740790 IC50 = 1128 nM T64969 C72PLS 141740792 IC50 = 16 nM T64969 CYU95H 141740794 IC50 = 203 nM T64969 C1Y4TJ 141740795 IC50 = 998 nM T64969 C62QXI 141740796 IC50 = 20 nM T64969 CDEX12 142518169 IC50 = 81.7 nM T64969 CCXG67 142735680 IC50 = 6 nM T64969 CP17MF 142747584 IC50 = 23 nM T64969 CGRY21 142747612 IC50 = 46 nM T64969 CQ15DI 142747615 IC50 = 38.7 nM T64969 C9THY0 145314346 IC50 = 257 nM T64969 CMHX97 145331319 IC50 = 1.4 nM T64969 CVID46 145331320 IC50 = 68 nM T64969 CW1P9K 145331325 IC50 = 81 nM T64969 CDB9Y1 145331327 IC50 = 2.5 nM T64969 CG6V5Q 145331334 IC50 = 17 nM T64969 CGPH07 145331338 IC50 = 4.7 nM T64969 C6C5DF 145331339 IC50 = 0.6 nM T64969 CXCO76 145331341 IC50 = 1.3 nM T64969 CO9P7G 145351804 IC50 > 1000 nM T64969 C6VB3O 145925651 IC50 >= 5000 nM T64969 C29XUO 145945978 IC50 > 1000 nM T64969 C91UGF 145946092 IC50 = 39 nM T64969 C4HB8M 145949394 IC50 = 812 nM T64969 CB3Z1W 145949428 IC50 = 8.7 nM T64969 CTR3F0 145949484 IC50 = 4 nM T64969 CK4N8D 145951329 IC50 = 71 nM T64969 C9TJ8F 145951621 IC50 = 174.5 nM T64969 CH8K2T 145952204 IC50 = 4100 nM T64969 CM3CX8 145952650 IC50 = 890 nM T64969 CKRP30 145952676 IC50 = 110 nM T64969 C8V4MP 145952681 IC50 = 865 nM T64969 CNI31W 145952990 IC50 = 5 nM T64969 COA5Y3 145953378 IC50 > 1000 nM T64969 CN4Q7F 145953551 IC50 = 37 nM T64969 CT53JG 145953604 IC50 = 32 nM T64969 CMH8O2 145953998 IC50 = 34 nM T64969 C89RPH 145954372 IC50 > 1000 nM T64969 CBY18Z 145954422 IC50 = 32 nM T64969 CW2OE8 145954892 IC50 > 1000 nM T64969 CFB43Y 145956534 IC50 = 17 nM T64969 C5VSC7 145956704 IC50 = 5400 nM T64969 C2V8DA 145957160 IC50 > 1000 nM T64969 CA3E2C 145957992 IC50 = 162 nM T64969 C42ZQH 145958534 IC50 > 1000 nM T64969 CXWH23 145958592 IC50 > 1000 nM T64969 CJE35T 145958671 IC50 = 45.4 nM T64969 C2IHF1 145960158 IC50 = 3350 nM T64969 CV57UK 145960288 IC50 = 16.4 nM T64969 C9R0TU 145960317 IC50 = 240 nM T64969 CC7ZP1 145960400 IC50 = 1.7 nM T64969 C4D2AW 145962014 IC50 = 4.5 nM T64969 CJT41L 145962084 IC50 > 10000 nM T64969 C1R6UI 145963124 IC50 = 29 nM T64969 CICN74 145963796 IC50 = 16970 nM T64969 CRMN13 145963949 Ki = 1360 nM T64969 C9E0LZ 145964191 IC50 = 3900 nM T64969 C2JXB0 145964277 IC50 = 500 nM T64969 C4K6RY 145964618 IC50 = 100 nM T64969 CJYQ32 145964655 IC50 = 595.4 nM T64969 C0KJR5 145964906 IC50 = 650 nM T64969 CI52HO 145965123 IC50 = 675 nM T64969 CN41TJ 145965367 IC50 > 1000 nM T64969 CLM8E6 145965506 IC50 = 9350 nM T64969 C3ZD2W 145965608 IC50 = 3870 nM T64969 CI1UV7 145965620 Ki = 680 nM T64969 CO7IH0 145965741 IC50 = 940 nM T64969 CTQ9S5 145965923 IC50 = 6980 nM T64969 C7YM1B 145966210 IC50 = 31.8 nM T64969 CP2MX0 145966312 IC50 = 2400 nM T64969 C3YGN7 145966332 Ki = 810 nM T64969 CHY74R 145966422 Ki = 930 nM T64969 CZ38PG 145966502 Ki = 230 nM T64969 C8UWY5 145966767 IC50 = 78 nM T64969 C5L7VC 145966803 IC50 = 34.8 nM T64969 CQE9M5 145966810 IC50 > 10000 nM T64969 C0G8ED 145966828 IC50 > 1000000 nM T64969 C4LHS5 145967074 Ki = 140 nM T64969 C4OD9Q 145967187 IC50 = 1.3 nM T64969 CS7CR2 145967258 Ki = 164 nM T64969 CDW83M 145967332 IC50 = 267.6 nM T64969 COZA32 145967334 Ki = 170 nM T64969 CM41TV 145967355 IC50 = 82.6 nM T64969 CUE4K8 145967670 IC50 = 3.5 nM T64969 C7NJ9Q 145967774 IC50 = 2140 nM T64969 CDNC31 145967951 IC50 > 500 nM T64969 CA0IB1 145967983 IC50 = 22330 nM T64969 CJO79P 145968146 IC50 = 24.2 nM T64969 C5E8ZK 145968310 IC50 > 1000 nM T64969 CM7HI4 145968374 IC50 = 2.692 nM T64969 C6UAM8 145968450 IC50 = 1230 nM T64969 C4RX3Q 145968531 IC50 = 49 nM T64969 C8BH4I 145968555 IC50 = 3.2 nM T64969 CU5HJ8 145968616 IC50 = 4.2 nM T64969 C2J0VU 145968689 Ki = 2050 nM T64969 CHAU61 145968737 IC50 > 1000 nM T64969 C9IMB1 145968764 IC50 = 2.3 nM T64969 CWJ12M 145969155 IC50 > 10000 nM T64969 C2HN8R 145969194 IC50 > 1000 nM T64969 C0GDV8 145969399 IC50 = 249.1 nM T64969 C1N0GM 145969603 IC50 = 842.3 nM T64969 CK82QG 145969816 IC50 = 409 nM T64969 CVXS26 145969908 IC50 = 529 nM T64969 CX4C6R 145970163 IC50 = 270 nM T64969 CTD6N0 145970346 IC50 = 510 nM T64969 C9ZO3X 145970379 IC50 = 28 nM T64969 CXE6W9 145970478 IC50 = 3.9 nM T64969 C1C6YP 145970679 IC50 = 5.1 nM T64969 C8NK3O 145970839 IC50 = 596 nM T64969 CON74U 145970883 IC50 = 18 nM T64969 C8BKZ3 145971291 IC50 = 98 nM T64969 CQ4FP9 145971558 IC50 = 6020 nM T64969 CAV7I1 145971580 IC50 = 0.9 nM T64969 CSJ0X9 145971962 IC50 = 60 nM T64969 C5G7ZX 145972214 IC50 > 1000 nM T64969 CW8UY6 145972402 Ki = 330 nM T64969 CH18WC 145972585 IC50 = 5640 nM T64969 CVQP05 145972782 IC50 = 39 nM T64969 CKY02W 145972834 IC50 = 1160 nM T64969 CKQ46V 145972976 Ki = 110 nM T64969 CH5E2D 145973277 IC50 > 1000000 nM T64969 CM21LZ 145973281 IC50 > 1000 nM T64969 CWP85Z 145973302 IC50 > 1000 nM T64969 C64GAI 145973339 IC50 = 3250 nM T64969 CH5IM9 145973468 IC50 = 260 nM T64969 CFZX58 145973489 IC50 = 9760 nM T64969 CN6JG9 145973510 IC50 = 8070 nM T64969 CTPQ06 145973553 Ki = 2740 nM T64969 CIKF18 145973791 Ki = 320 nM T64969 CHGD35 145974340 IC50 = 72 nM T64969 CIWU86 145974353 Ki = 110 nM T64969 CQH3G7 145974613 IC50 = 1590 nM T64969 CXRY95 145974888 IC50 = 6900 nM T64969 C5JR6E 145974924 Ki = 2 nM T64969 CE35TV 145975018 IC50 = 1700 nM T64969 CX4S7R 145975100 IC50 = 9040 nM T64969 CI4JO0 145975282 IC50 = 0.9 nM T64969 C74TYP 145975351 IC50 > 100000 nM T64969 CSE6N1 145975386 IC50 = 190.6 nM T64969 C5HB7J 145975494 IC50 > 1000000 nM T64969 CZ98JF 145975496 IC50 = 1070 nM T64969 CCUX93 145975528 IC50 = 230 nM T64969 C2WK8V 145975646 IC50 = 2.1 nM T64969 C6MX1J 145976050 IC50 = 8550 nM T64969 C28GAM 145976336 IC50 = 1410 nM T64969 C3LR4O 145976442 IC50 = 2.4 nM T64969 C1IUN8 145976637 IC50 = 215.4 nM T64969 CI7S4L 145976764 Ki = 400 nM T64969 CH64BI 145976972 IC50 = 9970 nM T64969 CD82JO 145977064 IC50 = 3070 nM T64969 CG57KO 145977147 IC50 = 13 nM T64969 CX41WF 145977261 IC50 = 3800 nM T64969 C69INU 145977311 Ki = 3590 nM T64969 C7WZG3 145977617 IC50 = 14010 nM T64969 CMK7P9 145977756 Ki = 183 nM T64969 C15XGN 145977927 Ki = 80 nM T64969 C46QAV 145977992 Ki = 2520 nM T64969 C71TVY 145978029 IC50 = 51.9 nM T64969 C6JB8T 145978055 IC50 = 24.7 nM T64969 C81QRF 145978122 IC50 = 1.1 nM T64969 CXC9F7 145978377 IC50 = 900 nM T64969 CT1QE0 145978442 IC50 = 6070 nM T64969 C6JBH1 145978562 Ki = 940 nM T64969 CRCM82 145978681 IC50 = 51.3 nM T64969 C5IVB9 145978838 Ki = 161 nM T64969 CCT8N6 145978865 IC50 = 102 nM T64969 CM2NU5 145978997 IC50 = 15.3 nM T64969 CTA34O 145979089 IC50 = 23 nM T64969 C2D4CA 145979249 IC50 > 100 nM T64969 C5TP2U 145979643 IC50 = 45000 nM T64969 CE31VG 145979714 IC50 > 10000 nM T64969 CN7KH0 145979764 IC50 = 1.5 nM T64969 C4X8LC 145979928 IC50 > 1000000 nM T64969 CT9A2R 145980005 IC50 = 100.5 nM T64969 CV60SM 145980007 IC50 = 0.8 nM T64969 C9QFA1 145980052 IC50 = 21.4 nM T64969 CU05GX 145980058 IC50 = 0.7 nM T64969 CZEK06 145980063 IC50 = 3.2 nM T64969 C0P7JL 145980218 IC50 = 0.7 nM T64969 C4BM0U 145980284 IC50 = 22.4 nM T64969 CNFJ75 145980559 IC50 > 1000000 nM T64969 C5LIK2 145980611 IC50 = 1409 nM T64969 C1A5PW 145980662 IC50 = 27 nM T64969 CL19AW 145980663 IC50 = 0.4 nM T64969 CVRB57 145980676 IC50 = 0.6 nM T64969 COI8B7 145981029 IC50 = 9 nM T64969 C8FRT3 145981115 IC50 = 27 nM T64969 C4J9SC 145981182 IC50 = 105 nM T64969 CU67FB 145981262 IC50 = 2.7 nM T64969 C72RDL 145981281 IC50 = 46 nM T64969 CP67EO 145981349 IC50 = 68 nM T64969 CVO6T8 145981395 IC50 = 592.1 nM T64969 CSW6P0 145981487 IC50 = 1182 nM T64969 CCD7Y3 145981564 IC50 = 7200 nM T64969 C47TVC 145981655 IC50 = 1500 nM T64969 CLX91B 145981733 IC50 = 47.1 nM T64969 C64FYE 145981880 IC50 = 0.7 nM T64969 C1H5JE 145982613 IC50 = 52110 nM T64969 CC12YA 145982666 IC50 = 6.4 nM T64969 CF4BO8 145982785 IC50 = 4 nM T64969 CM6ZS7 145982824 IC50 = 3.1 nM T64969 CUN92A 145982933 IC50 = 21.5 nM T64969 C35FMR 145983116 IC50 > 100 nM T64969 C0YFS6 145983170 IC50 > 100 nM T64969 CF28AU 145983389 IC50 = 10.1 nM T64969 C48ZXP 145983545 IC50 > 100 nM T64969 C4QE7K 145983757 IC50 = 1200 nM T64969 CD5L8O 145983778 IC50 > 200 nM T64969 CM8Z7V 145984082 IC50 > 100 nM T64969 C1DM4I 145984486 IC50 = 1900 nM T64969 COPW70 145984516 IC50 = 1400 nM T64969 CYG42V 145984818 IC50 > 200 nM T64969 CLVN80 145984870 IC50 = 38730 nM T64969 CFS7D5 145984941 IC50 > 200 nM T64969 C05IMJ 145984942 IC50 = 7.1 nM T64969 CPHN84 145985403 IC50 = 467 nM T64969 CS9C8J 145986155 IC50 > 200 nM T64969 CY5NX4 145986312 IC50 = 1 nM T64969 C2T4PK 145986404 IC50 = 5600 nM T64969 CV45JH 145986520 IC50 = 754 nM T64969 C8EUL5 145986728 IC50 = 2700 nM T64969 CB80EO 145986808 IC50 > 1000 nM T64969 CCJ19R 145986823 IC50 = 2.6 nM T64969 CGI48S 145986878 IC50 = 0.3 nM T64969 CB48CA 145986981 IC50 = 0.7 nM T64969 C1Y5MO 145987062 IC50 = 632.8 nM T64969 CRKD41 145987099 IC50 = 901 nM T64969 CAE5G0 145987157 IC50 > 1000000 nM T64969 CJ2A5I 145987445 IC50 = 951 nM T64969 CU96RK 145987761 IC50 = 944 nM T64969 CF6KO7 145987807 IC50 = 1 nM T64969 C0MI7K 145988025 IC50 = 21 nM T64969 C7A4WK 145988274 IC50 = 47.7 nM T64969 C3N8OJ 145988373 IC50 = 288 nM T64969 C4FWV5 145988395 IC50 = 1931 nM T64969 CDVL79 145988898 IC50 = 33 nM T64969 CZ1VH0 145988939 IC50 = 94.7 nM T64969 C9BX4U 145988956 IC50 > 10000 nM T64969 CP9N1M 145989301 IC50 = 205 nM T64969 C74MSY 145989401 IC50 = 17 nM T64969 C2VA1T 145989472 IC50 = 1700 nM T64969 C2B0LS 145989721 IC50 = 62.5 nM T64969 CB13UV 145989878 IC50 = 0.8 nM T64969 CWI75O 145990017 IC50 = 120 nM T64969 C2PBJ5 145990245 IC50 = 112 nM T64969 CH17ZV 145990291 IC50 = 13.4 nM T64969 CX4YJ5 145990338 IC50 = 0.71 nM T64969 CTC0L2 145990413 IC50 = 60 nM T64969 CE1QB4 145990507 IC50 = 229 nM T64969 CNQ91H 145990537 IC50 = 26 nM T64969 C9Q6XC 145990684 IC50 = 0.7 nM T64969 COS6Z7 145990801 IC50 = 24.8 nM T64969 C1J5IX 145990848 IC50 > 1000000 nM T64969 CRS5P2 145991103 IC50 = 1.4 nM T64969 CD79LS 145991130 IC50 = 9800 nM T64969 C0XBV2 145991309 IC50 = 752 nM T64969 C5KB0A 145991472 IC50 > 1000000 nM T64969 COU0E6 145991881 IC50 = 91.7 nM T64969 C2CBQ4 145992100 IC50 = 751 nM T64969 C4YUL3 145992531 IC50 = 96.6 nM T64969 CZP7Y0 145992597 IC50 = 1229 nM T64969 C4A2UC 145992646 IC50 = 70 nM T64969 C2FQG8 145992679 IC50 = 2800 nM T64969 CO41PW 145992706 IC50 = 792 nM T64969 CNC69T 145992844 IC50 > 100000 nM T64969 C0C4ZD 145993006 IC50 = 11 nM T64969 CWK20P 145993042 IC50 = 108 nM T64969 C7Q6NU 145993198 IC50 = 933 nM T64969 CW8E2A 145993359 IC50 = 1 nM T64969 C85KQX 145993400 IC50 = 1.2 nM T64969 CZ6OC9 145993414 IC50 = 37 nM T64969 CS8UQ5 145994037 IC50 = 8.6 nM T64969 C6B3TD 146014465 IC50 = 13 nM T64969 CQNH23 146180715 IC50 = 9.3 nM T64969 C6YC0B 146180716 IC50 = 179.6 nM T64969 CJU8M7 146180717 IC50 = 2.2 nM T64969 CS6FR4 146180753 IC50 = 19.2 nM T64969 CK18RY 146180803 IC50 = 37.1 nM T64969 CS2Q4N 146182117 IC50 = 7.9 nM T64969 CF06AW 146197277 IC50 > 20000 nM T64969 CRP36X 146197294 IC50 > 20000 nM T64969 COJM12 146197324 IC50 > 20000 nM T64969 C8S7QZ 146197334 IC50 > 20000 nM T64969 C9MO7E 146197361 IC50 > 20000 nM T64969 CW9Y5K 146197370 IC50 > 20000 nM T64969 CO27GX 146197371 IC50 > 20000 nM T64969 CFV2O7 146197389 IC50 > 20000 nM T64969 C1X2MP 146197393 IC50 > 20000 nM T64969 C0CN9F 146197408 IC50 > 20000 nM T64969 CO1F2N 146197447 IC50 > 20000 nM T64969 CBJR67 146197457 IC50 > 20000 nM T64969 CG86IF 146197468 IC50 > 20000 nM T64969 CD7Y8E 146212989 IC50 > 20000 nM T64969 CBM7C5 146773032 IC50 = 12450 nM T64969 CP81CX 146832100 IC50 = 76 nM T64969 C9D1EH 147117461 IC50 = 18690 nM T64969 C8I1HV 147384518 IC50 = 16180 nM T64969 C7DYK4 147709549 IC50 = 18260 nM T64969 CIT79C 148291912 IC50 = 9570 nM T64969 C2U0SJ 148390225 IC50 = 26970 nM T64969 CJ23ZE 148637488 IC50 = 15360 nM T64969 CVL49H 149513019 IC50 = 22850 nM T64969 CR20QN 149611945 IC50 = 39 nM T64969 CYN8L2 152157601 IC50 > 10000 nM T64969 CSE96B 152685456 IC50 = 315 nM T64969 CFKU39 152790957 IC50 = 30450 nM T64969 CS7Q1E 152878273 IC50 = 52 nM T64969 CV41DF 153011787 IC50 = 25410 nM T64969 C60JPV 155166360 IC50 = 149 nM T64969 CL41OU 155183985 IC50 = 2 nM T64969 C90HPT 155338585 IC50 = 31 nM T64969 CP5NX6 155338590 IC50 = 12 nM T64969 CRC8D2 155489850 IC50 = 2200 nM T64969 CZ4V5U 155510439 IC50 > 1000 nM T64969 C03YFP 155510706 IC50 = 38 nM T64969 C5Z7GK 155511049 IC50 = 4.95 nM T64969 CDR04S 155511317 IC50 = 15 nM T64969 CQI50K 155511379 IC50 = 81 nM T64969 CY7X0V 155511571 IC50 = 28.2 nM T64969 CWZ2S8 155511862 IC50 = 4.3 nM T64969 CE10PX 155512047 IC50 = 5 nM T64969 CL4B2M 155512535 IC50 = 147 nM T64969 CKR0P6 155512805 IC50 = 25 nM T64969 C81YCJ 155513061 IC50 = 70 nM T64969 C9NT2X 155513114 IC50 = 30 nM T64969 C2MD1Q 155513187 IC50 > 10000 nM T64969 CQ3XH4 155513485 IC50 = 500 nM T64969 COZ61S 155513553 IC50 = 46.52 nM T64969 CU12GD 155513666 IC50 = 10580 nM T64969 C17INE 155513714 IC50 = 397 nM T64969 CI78ZM 155513927 IC50 = 10 nM T64969 C7SK0E 155513959 IC50 = 40.6 nM T64969 C1XNV5 155513991 IC50 = 9 nM T64969 CHG6K2 155514100 IC50 = 320 nM T64969 CBP9L6 155514128 IC50 = 450 nM T64969 CKN04R 155514224 IC50 = 34 nM T64969 C3EXJ1 155514609 IC50 = 52.6 nM T64969 C7SPR0 155514679 IC50 = 111 nM T64969 CD46IN 155514865 IC50 = 61 nM T64969 C7YEN3 155514902 IC50 = 0.87 nM T64969 C7AMX8 155514903 IC50 > 3000 nM T64969 C1K3OA 155515133 IC50 = 710 nM T64969 CDAL34 155515494 IC50 = 844 nM T64969 CT2C5D 155515585 IC50 = 54.69 nM T64969 CC7N4A 155515743 IC50 = 4520 nM T64969 CU76NE 155516227 IC50 = 24130 nM T64969 CI23DH 155516489 IC50 = 1257 nM T64969 CR2D9I 155516959 IC50 = 16 nM T64969 C8GX0B 155517202 IC50 = 2700 nM T64969 C4D1WA 155517369 IC50 = 4750 nM T64969 C36ZMS 155518518 IC50 > 50000 nM T64969 C86HPW 155518524 IC50 = 10000 nM T64969 CJ0O8S 155518727 IC50 = 1248 nM T64969 CPTF82 155518915 IC50 = 79 nM T64969 CH42VE 155518994 IC50 = 2459 nM T64969 CG4C2D 155519085 IC50 = 500 nM T64969 C3VTM7 155519139 IC50 = 400 nM T64969 C0BZ6I 155519249 IC50 = 416 nM T64969 CTS0J7 155519458 IC50 = 400 nM T64969 CE83DJ 155519522 IC50 = 1259 nM T64969 C3NA2I 155519537 IC50 > 1000 nM T64969 CC8BO2 155519579 IC50 = 1700 nM T64969 CR68FM 155519610 IC50 > 1000 nM T64969 C9HEY1 155519702 IC50 = 26150 nM T64969 CYO23E 155519705 IC50 = 32.5 nM T64969 CBY13X 155519739 EC50 = 2 nM T64969 CNU28S 155519814 IC50 > 1000 nM T64969 CQAN74 155519895 IC50 = 105 nM T64969 C01HMD 155519991 IC50 = 239 nM T64969 C1X6YD 155520212 IC50 = 1322 nM T64969 C6K8NG 155520384 IC50 = 499 nM T64969 COQ7U0 155520571 EC50 = 4 nM T64969 C98UXO 155520734 IC50 = 0.34 nM T64969 C3UAF7 155521257 IC50 = 65.34 nM T64969 C9FVT0 155521452 IC50 = 123.2 nM T64969 CF93WQ 155521654 IC50 = 395 nM T64969 CWVX73 155522179 IC50 = 54.99 nM T64969 C8ZDA3 155522205 IC50 = 562 nM T64969 CNIR83 155522516 IC50 = 224.1 nM T64969 CB50GK 155522849 IC50 = 43.56 nM T64969 CHRT30 155522905 IC50 = 20 nM T64969 CI65WG 155523218 IC50 = 227.9 nM T64969 CES5L2 155523448 IC50 = 65.2 nM T64969 CNLC48 155523465 IC50 = 23.4 nM T64969 C2NQV1 155523617 IC50 = 421 nM T64969 CZ6ES5 155524096 IC50 = 0.5872 nM T64969 CA9YF3 155524153 IC50 = 38 nM T64969 C5EZR1 155524215 IC50 = 68 nM T64969 CD7ZH8 155524226 IC50 > 20000 nM T64969 C3TF9E 155524436 IC50 = 120.7 nM T64969 C5R8SL 155524645 IC50 > 20000 nM T64969 CH6FQ9 155524667 IC50 = 4300 nM T64969 CJBE61 155524820 IC50 = 6300 nM T64969 C0COA7 155525819 IC50 = 62 nM T64969 CJ35GA 155525934 IC50 = 4240 nM T64969 CRT67D 155526236 IC50 = 8.7 nM T64969 CFAS17 155526847 IC50 = 13 nM T64969 CE3OH1 155527121 IC50 = 138 nM T64969 C3GNP6 155527669 IC50 = 2.5 nM T64969 C8I3SW 155527677 IC50 = 12 nM T64969 CQLF39 155527847 IC50 = 16.43 nM T64969 C3HP8E 155527851 IC50 = 18 nM T64969 CF39US 155528086 IC50 = 421 nM T64969 C72HJM 155528259 IC50 > 1000 nM T64969 C47YUC 155528358 IC50 > 20000 nM T64969 C9P2NQ 155528441 IC50 = 8770 nM T64969 CHI54P 155529236 IC50 = 617 nM T64969 C10JWF 155529388 IC50 = 14 nM T64969 CFKV53 155529663 IC50 = 22.7 nM T64969 CW9OC4 155529736 IC50 = 37.1 nM T64969 CN40AE 155529739 IC50 = 700 nM T64969 CUXA18 155529935 IC50 = 903 nM T64969 CLJ5T9 155529954 IC50 = 18.54 nM T64969 CU96GQ 155529955 IC50 = 64 nM T64969 CL0US4 155530459 IC50 = 2.3 nM T64969 CQLV68 155530541 IC50 = 1600 nM T64969 C6VQ0W 155530641 IC50 > 1000 nM T64969 C2WCU6 155530774 IC50 = 1048 nM T64969 C3N4UG 155530777 IC50 = 1771 nM T64969 CX7I1V 155531079 IC50 = 765 nM T64969 CWO98B 155531773 IC50 = 9 nM T64969 CVBK76 155531967 IC50 > 1000 nM T64969 C8HDO1 155532442 IC50 = 3 nM T64969 CGVZ73 155532854 IC50 > 1000 nM T64969 C3D5JZ 155533027 IC50 = 177 nM T64969 CJ6T5H 155533092 IC50 = 12 nM T64969 CNQP76 155533136 IC50 > 1000 nM T64969 CQFC65 155533189 IC50 = 2400 nM T64969 C7OX2W 155533223 IC50 = 19.97 nM T64969 CNGX84 155533637 IC50 = 2750 nM T64969 C5UQG3 155534199 IC50 = 8.7 nM T64969 C1NGV5 155534208 IC50 = 499 nM T64969 C4TRF0 155534357 IC50 = 3660 nM T64969 C3J4OM 155534528 IC50 > 20000 nM T64969 CM0U3I 155534552 IC50 > 1000 nM T64969 CEQJ52 155534874 IC50 > 1000 nM T64969 C6QX2V 155534940 IC50 = 31.7 nM T64969 CMH2J4 155535076 IC50 = 0.69 nM T64969 CD8TO7 155535214 IC50 = 15330 nM T64969 C3RWB0 155535296 IC50 = 31 nM T64969 CRI7V1 155535998 IC50 = 1753 nM T64969 C78MZC 155536330 IC50 = 2 nM T64969 C6H7QE 155536433 IC50 = 83 nM T64969 CF0A9O 155536643 IC50 = 10 nM T64969 CBS75N 155536946 IC50 = 2800 nM T64969 C2CG1A 155537016 IC50 > 10000 nM T64969 C2SW1K 155537706 IC50 = 201 nM T64969 CP3AD2 155537718 IC50 = 81 nM T64969 CZNX25 155537733 IC50 = 234 nM T64969 CP8ZV6 155538283 IC50 = 4 nM T64969 C6Z7XO 155538664 IC50 = 2.213 nM T64969 C0IH1J 155539209 IC50 = 105.3 nM T64969 CEN71T 155539953 IC50 = 20.83 nM T64969 CC3IQ7 155540048 IC50 = 26 nM T64969 C1B0VO 155540273 IC50 = 4.3 nM T64969 CE46SL 155540854 IC50 = 4340 nM T64969 C5O4JM 155540856 IC50 = 23340 nM T64969 CX68YN 155541385 IC50 > 50000 nM T64969 CLY07P 155541605 IC50 > 150 nM T64969 CT02GE 155541767 IC50 = 598 nM T64969 CH10DU 155542091 IC50 = 654 nM T64969 CNR2X9 155542138 IC50 = 119.7 nM T64969 C7X2KJ 155542371 IC50 = 70 nM T64969 CP67JN 155542393 IC50 = 5.9 nM T64969 C02VLJ 155542715 IC50 = 4 nM T64969 CTQ9S4 155543012 IC50 = 1.4 nM T64969 CW73EO 155543439 IC50 = 38 nM T64969 C1VJH0 155543634 IC50 = 36840 nM T64969 C0JR1M 155544107 IC50 = 0.62 nM T64969 CUT37P 155544297 IC50 = 20 nM T64969 C5ZMA0 155544307 IC50 = 5004 nM T64969 CVG79N 155544855 IC50 = 3059 nM T64969 C1SMF6 155545153 IC50 = 133 nM T64969 CGE04I 155545288 IC50 = 820 nM T64969 CEJ3V2 155545290 IC50 = 56.1 nM T64969 C4H9XV 155545331 IC50 = 209 nM T64969 CCHK04 155545559 IC50 = 50.8 nM T64969 CPKS19 155545810 IC50 = 5 nM T64969 CN18UI 155545963 IC50 = 14 nM T64969 C46MQV 155546345 IC50 = 9 nM T64969 CJN15V 155546412 IC50 = 6.24 nM T64969 CSI83K 155546458 IC50 = 12.93 nM T64969 CAVB85 155546598 IC50 > 10000 nM T64969 CTBA51 155546884 IC50 = 6 nM T64969 CFA1X6 155546954 IC50 = 6.6 nM T64969 C10XPU 155547167 EC50 = 666 nM T64969 CN4PM8 155547174 IC50 = 1.15 nM T64969 C7SF2C 155547229 IC50 > 10000 nM T64969 CL8X7V 155547722 IC50 = 48.07 nM T64969 CFR63D 155547749 IC50 = 275.7 nM T64969 CGX7Z0 155548089 IC50 = 40 nM T64969 C60YKA 155548301 IC50 > 1000 nM T64969 CV54FM 155548416 IC50 = 6600 nM T64969 CE6M4K 155548572 IC50 = 174 nM T64969 CBN4M1 155548812 IC50 = 44 nM T64969 CZ7WR0 155549232 IC50 = 8 nM T64969 CNG4O3 155549841 IC50 = 2900 nM T64969 CL1E6U 155549934 IC50 = 27.92 nM T64969 CY6RU2 155549975 IC50 = 0.37 nM T64969 CV7S6N 155550199 IC50 = 4 nM T64969 C9J1MU 155550347 IC50 = 2 nM T64969 C93NWJ 155550657 IC50 = 148.8 nM T64969 C49SQG 155551406 IC50 = 23 nM T64969 C3UBY1 155551683 IC50 = 1128.9 nM T64969 CEDT28 155552106 IC50 = 26 nM T64969 CZ4J2P 155552610 IC50 > 1000 nM T64969 C0HUL3 155552710 IC50 = 1975 nM T64969 C2VNW3 155553566 IC50 = 52 nM T64969 CAC31S 155553712 IC50 = 2 nM T64969 CGVU70 155554426 IC50 = 4710 nM T64969 C5MAK6 155554594 IC50 = 45.2 nM T64969 CJ0G2I 155554715 IC50 = 35 nM T64969 CD9M1F 155554777 IC50 = 273 nM T64969 C2T1XS 155554878 IC50 = 591 nM T64969 C1FJ5D 155555800 IC50 > 20000 nM T64969 CT6S9X 155555827 IC50 = 120.2 nM T64969 CWDR07 155555935 IC50 = 15630 nM T64969 C3F8YQ 155556804 IC50 = 368 nM T64969 CX96CQ 155556857 IC50 = 32.61 nM T64969 C5KSJ1 155556978 IC50 = 93 nM T64969 C4BH8P 155557234 IC50 = 12 nM T64969 CQ9GK2 155557533 IC50 = 27 nM T64969 C2LWI3 155557949 IC50 = 157 nM T64969 CARD46 155557959 IC50 = 197 nM T64969 CZD71I 155558249 IC50 = 3.11 nM T64969 CC8R3X 155558455 IC50 = 188 nM T64969 C10OFJ 155558962 IC50 = 0.6 nM T64969 CPAV79 155559005 IC50 > 3000 nM T64969 C89XOB 155559201 IC50 = 5.6 nM T64969 C2Q8OK 155559257 IC50 = 105 nM T64969 CL3JM7 155559534 IC50 = 153.5 nM T64969 C1OI5K 155559863 IC50 > 1000 nM T64969 CBA35K 155559950 IC50 = 77 nM T64969 C51IBQ 155560019 IC50 = 937 nM T64969 CXZ74V 155560104 IC50 > 150 nM T64969 CCD34P 155560610 IC50 = 3200 nM T64969 CT2XQ0 155561007 IC50 = 215 nM T64969 C8J0IZ 155561310 IC50 > 1000 nM T64969 CM3JG6 155561359 IC50 = 2 nM T64969 C6N1KS 155561750 IC50 = 146.2 nM T64969 CES3Q5 155561884 IC50 = 1200 nM T64969 CT7UJ9 155562064 IC50 = 104 nM T64969 CFI4C8 155562148 IC50 = 85 nM T64969 CC5F3I 155562216 IC50 = 84 nM T64969 CTF4Z2 155562466 IC50 > 1000 nM T64969 C87PUX 155562472 IC50 = 107.2 nM T64969 CNDL07 155562495 IC50 = 141 nM T64969 C1VCU9 155562538 IC50 = 33.31 nM T64969 C1ZX4J 155563060 IC50 > 1000 nM T64969 C9V5HT 155563732 IC50 = 142.7 nM T64969 C9L6WZ 155563761 IC50 > 150 nM T64969 C7XK2B 155564005 IC50 = 118.6 nM T64969 CS37KE 155564015 IC50 = 12000 nM T64969 CAC85T 155564156 IC50 > 3000 nM T64969 CT53XC 155564242 IC50 = 1 nM T64969 CU7Z0H 155564272 IC50 = 3.7 nM T64969 CLPY65 155564381 IC50 = 326 nM T64969 CY9BN3 155564537 IC50 = 11 nM T64969 C3F6ML 155564606 IC50 = 2160 nM T64969 CQ1N7J 155564622 IC50 = 38.5 nM T64969 CY1KP0 155564719 IC50 = 92 nM T64969 CBS5F3 155564756 IC50 = 8 nM T64969 C0ZWD9 155565268 IC50 = 302 nM T64969 C0UG5P 155565835 IC50 > 150 nM T64969 CA36ST 155565961 IC50 = 19 nM T64969 CWAF51 155566440 IC50 = 12 nM T64969 C3G5LQ 155566848 IC50 > 1000 nM T64969 C04KYS 155566973 IC50 = 8.3 nM T64969 CZC73X 155567166 IC50 = 2880 nM T64969 CUB2J0 155567333 IC50 = 1400 nM T64969 C5AO3Q 155567359 IC50 = 60 nM T64969 C6LI4S 155567410 IC50 = 12.57 nM T64969 CQS81I 155568841 IC50 = 108 nM T64969 CMNZ49 155569055 IC50 > 2000 nM T64969 CGU74Q 155569301 IC50 = 150 nM T64969 C1IC3A 14862543 IC50 = 40000 nM T64969 CLQ6F4 14862545 IC50 = 7000 nM T64969 D00ATA 5908088 IC50 > 100000 nM T64969 D00ERW 44444843 Ki > 1803 nM T64969 D00GVV 5329155 IC50 > 100000 nM T64969 D00HVA 11624601 Ki > 1800 nM T64969 D00LRC 10422592 IC50 > 20000 nM T64969 D00RBV 10445611 IC50 > 25000 nM T64969 D00RIX 5280443 IC50 = 30 ug.mL-1 T64969 D00TBD 10461815 IC50 = 3800 nM T64969 D00TJF 11807783 IC50 = 3.38 nM T64969 D00TZD 2776 IC50 = 0.37 nM T64969 D00VZA 5328763 IC50 = 1000 nM T64969 D00WZG 44442168 IC50 = 15 nM T64969 D01NTW 5328768 Ki = 3500 nM T64969 D01OKF 46207013 IC50 = 580 nM T64969 D01RHR 71519693 IC50 = 11 nM T64969 D01UYS 11778521 IC50 > 20000 nM T64969 D01VFR 4708 IC50 = 0.08 nM T64969 D01WXV 44442181 IC50 = 15 nM T64969 D01WYI 9995195 IC50 = 0.42 nM T64969 D02BUW 2061 Ki = 1000 nM T64969 D02BXJ 46864270 IC50 = 736 nM T64969 D02CUF 10424517 IC50 > 20000 nM T64969 D02KVB 5328804 IC50 = 125 nM T64969 D02NNT 53232451 IC50 > 10000 nM T64969 D02RIG 5328755 IC50 = 7000 nM T64969 D02ZRO 735125 IC50 = 27 nM T64969 D03ATU 4707 IC50 = 0.008 nM T64969 D03BJB 9549299 IC50 = 21 nM T64969 D03CVQ 44442182 IC50 = 5 nM T64969 D03EHM 24905142 IC50 = 260 nM T64969 D03HLH 44331231 IC50 = 70 nM T64969 D03MUZ 17759555 IC50 = 1800 nM T64969 D03OKV 9844320 IC50 > 1000 nM T64969 D03XDN 4709 IC50 = 0.1 nM T64969 D04FNY 25195216 IC50 = 3480 nM T64969 D04HGN 2809539 IC50 = 6300 nM T64969 D04LXG 44442183 IC50 = 140 nM T64969 D04NGS 5330790 IC50 > 100000 nM T64969 D04PEI 11467730 IC50 > 50000 nM T64969 D04XNJ 4879 IC50 = 2700 nM T64969 D05ARF 5328077 IC50 = 578 nM T64969 D05EDW 10085862 IC50 > 20000 nM T64969 D05FFT 11566580 IC50 = 0.3 nM T64969 D05GBY 10242258 IC50 > 20000 nM T64969 D05QMN 44331083 IC50 = 2500 nM T64969 D05SNG 10398928 IC50 > 20000 nM T64969 D06BJG 71556703 IC50 = 7 nM T64969 D06HVH 54613583 IC50 > 10000 nM T64969 D06KSF 9549300 IC50 < 5000 nM T64969 D06LJL 9916282 IC50 = 800 nM T64969 D06LLF 10017166 IC50 > 20000 nM T64969 D06MCJ 9972296 IC50 > 20000 nM T64969 D06QWO 14824655 IC50 > 10 ug.mL-1 T64969 D06UEK 15984068 IC50 = 710 nM T64969 D06VNR 10085863 IC50 > 20000 nM T64969 D07CFT 10447210 IC50 > 20000 nM T64969 D07IHD 5328753 IC50 = 500 nM T64969 D07IHM 9823787 IC50 > 10000 nM T64969 D07JDY 10243001 IC50 > 20000 nM T64969 D07OCA 5330812 IC50 > 10000 nM T64969 D07OSK 6419834 IC50 > 100000 nM T64969 D07OXC 11650194 IC50 = 1700 nM T64969 D07SRX 9797919 IC50 = 7300 nM T64969 D07UYV 2857 IC50 = 0.006 nM T64969 D07ZWN 10060170 IC50 > 20000 nM T64969 D08JGS 11722903 IC50 > 20000 nM T64969 D08KWL 10402251 IC50 > 20000 nM T64969 D08LYB 5166 IC50 = 83 nM T64969 D08NQM 5289247 IC50 > 10000 nM T64969 D08RZB 11153014 IC50 = 5200 nM T64969 D08SUH 10336427 IC50 > 20000 nM T64969 D08WOG 9948853 IC50 = 20 nM T64969 D09HVH 135566652 IC50 > 10 nM T64969 D09LPL 5329103 IC50 = 3000 nM T64969 D09QBA 23378546 IC50 > 10000 nM T64969 D09TNR 9850161 IC50 > 10000 nM T64969 D09XIL 11396738 IC50 = 545 nM T64969 D0A0JL 2052 Ki = 11000 nM T64969 D0A1CM 5281855 IC50 = 690 nM T64969 D0A4XJ 5289418 IC50 > 100000 nM T64969 D0A6AA 10083695 IC50 > 20000 nM T64969 D0A6YP 9971060 IC50 > 20000 nM T64969 D0A9RM 5281804 IC50 = 4 ug.mL-1 T64969 D0AO6T 10402592 IC50 > 20000 nM T64969 D0AU0M 637542 Ki = 1000000 nM T64969 D0B4PH 2426 IC50 = 0.12 nM T64969 D0B8DE 135469328 IC50 = 5000 nM T64969 D0BU6T 354471 IC50 = 500 nM T64969 D0BW4G 10907042 IC50 > 30000 nM T64969 D0C1BE 10401378 IC50 > 20000 nM T64969 D0C2GE 67161540 IC50 = 137 nM T64969 D0C9KC 10850934 IC50 = 95 nM T64969 D0CF9B 10265642 IC50 > 20000 nM T64969 D0D2FC 2794188 IC50 = 5100 nM T64969 D0D5EW 5311104 IC50 = 390 nM T64969 D0D6DH 10125830 IC50 > 50000 nM T64969 D0D6MH 11617559 IC50 > 24000 nM T64969 D0D9PD 11656591 IC50 = 720 nM T64969 D0D9TU 3894 IC50 = 0.004 ug.mL-1 T64969 D0DF3Z 2808977 IC50 = 4.6 nM T64969 D0EE6A 6398883 IC50 > 1000 nM T64969 D0EH6L 10360970 IC50 = 4500 nM T64969 D0EU1R 46215815 IC50 > 10000 nM T64969 D0EW3L 5281222 IC50 = 8000 nM T64969 D0F6FZ 10494722 IC50 = 90 nM T64969 D0FH3M 18770833 IC50 = 4000 nM T64969 D0G0KN 9882618 IC50 > 20000 nM T64969 D0G0ZQ 10468421 IC50 > 20000 nM T64969 D0G3SZ 6918469 IC50 = 9.8 ug.mL-1 T64969 D0G3TK 5280863 IC50 = 3 ug.mL-1 T64969 D0G4HR 14862522 IC50 = 1000 nM T64969 D0G6SA 10422972 IC50 > 20000 nM T64969 D0G8GA 350901 IC50 = 15000 nM T64969 D0G9KD 5328245 IC50 = 0.003 nM T64969 D0GN3E 10243546 IC50 > 20000 nM T64969 D0GW4Q 5330524 IC50 = 380 nM T64969 D0H2CM 135565635 IC50 = 4400 nM T64969 D0H3UI 2063 Ki > 400000 nM T64969 D0H4JB 11778467 IC50 > 20000 nM T64969 D0HD2G 4788 IC50 = 25000000 nM T64969 D0HE0E 5941540 IC50 > 100000 nM T64969 D0HM5W 5328042 IC50 = 0.78 nM T64969 D0I0GL 10039460 IC50 > 20000 nM T64969 D0I7RA 11696664 IC50 = 131 nM T64969 D0IR5I 135453851 IC50 = 500 nM T64969 D0J5SK 5328819 IC50 = 2700 nM T64969 D0K2VO 44442165 IC50 = 14 nM T64969 D0K7GD 5328045 IC50 = 0.1 nM T64969 D0K9ON 10040402 IC50 > 20000 nM T64969 D0KF3N 10083699 IC50 > 20000 nM T64969 D0L0HG 766949 IC50 > 10000 nM T64969 D0L3FK 5289419 IC50 > 10000 nM T64969 D0L3SN 6439158 IC50 = 8800 nM T64969 D0L4HJ 5330462 IC50 = 5400 nM T64969 D0L8HO 2399 IC50 > 50000 nM T64969 D0M4SY 135440466 IC50 = 1600 nM T64969 D0M9QM 5327820 IC50 = 800 nM T64969 D0ME9B 46868971 IC50 > 10 nM T64969 D0N8TQ 10401956 IC50 < 1 nM T64969 D0NH7M 5328760 IC50 = 370 nM T64969 D0NS1S 5280442 IC50 = 40 ug.mL-1 T64969 D0O6OH 71553154 IC50 = 590 nM T64969 D0O9UR 638439 IC50 = 7900 nM T64969 D0P0RD 10065445 IC50 > 20000 nM T64969 D0P0WT 3139 IC50 > 10000 nM T64969 D0P2GE 18770812 IC50 = 5600 nM T64969 D0P3JW 447700 IC50 = 90 nM T64969 D0P6JS 11675054 IC50 > 10000 nM T64969 D0Q0YV 24944925 IC50 > 19952.62 nM T64969 D0Q3EW 9549303 IC50 > 10000 nM T64969 D0Q3GG 667601 Ki = 850 nM T64969 D0Q3NG 11715520 Ki > 1800 nM T64969 D0QC0W 9914412 IC50 = 110 nM T64969 D0QN6U 9806182 IC50 > 10000 nM T64969 D0RD5S 10355832 IC50 > 20000 nM T64969 D0S0RK 10680 IC50 = 50 ug.mL-1 T64969 D0S7IE 11658882 Ki > 1800 nM T64969 D0S9QP 44442180 IC50 = 26 nM T64969 D0S9YX 5280373 IC50 = 30 ug.mL-1 T64969 D0SJ2Q 10494 IC50 > 20000 nM T64969 D0SY2M 5281708 IC50 > 100 ug.mL-1 T64969 D0T9FQ 10061448 IC50 > 10000 nM T64969 D0U3WQ 9817165 IC50 > 30000 nM T64969 D0U6WB 2427 IC50 = 0.025 nM T64969 D0UN9O 3385203 IC50 >= 10000 nM T64969 D0V8QI 10331922 IC50 > 20000 nM T64969 D0V9EN 689043 Ki = 400000 nM T64969 D0W1BE 638437 IC50 = 10000 nM T64969 D0W6CE 10644450 IC50 = 10500 nM T64969 D0W7IN 10083051 IC50 > 20000 nM T64969 D0W9BF 9903563 IC50 > 20000 nM T64969 D0WW8M 10446889 IC50 > 20000 nM T64969 D0X4IO 5350 IC50 = 9000 nM T64969 D0X4UE 10220590 IC50 = 1000 nM T64969 D0XS9E 5330535 IC50 > 30000 nM T64969 D0Y2AM 5328038 IC50 = 355 nM T64969 D0YE1X 9927943 IC50 > 10000 nM T64969 D0YZ7H 9797370 IC50 > 100000 nM T64969 D0Z4HV 10354294 IC50 > 10000 nM T64969 D0Z7TM 22273644 IC50 > 1000 nM T64969 D0ZH1U 2051 IC50 = 120 nM T64969 D0ZT9D 6450172 IC50 = 1600 nM T04497 CNX67F 11951384 Ki = 1610 nM T04497 C17YPD 25138121 Ki = 23422 nM T04497 C0ZH5A 25138122 Ki = 71162 nM T95286 CSLT92 25138851 IC50 = 37400 nM T95286 C4P2XC 25140736 IC50 = 136000 nM T95286 C7CXU9 53317637 IC50 = 171000 nM T95286 CKE7U4 53318681 IC50 = 9270 nM T95286 CFUB60 53322630 IC50 = 164000 nM T95286 CMYR56 53323963 IC50 = 16600 nM T95286 C03QAM 56660019 IC50 = 272000 nM T95286 CA79VN 56660021 IC50 = 79 nM T95286 C42IUZ 56663487 IC50 = 610 nM T95286 CD84IP 56663489 IC50 = 640 nM T95286 CLYS24 56664906 IC50 = 9 nM T95286 CBI5N2 56666910 IC50 = 1200 nM T95286 CV3HX5 56668531 IC50 = 7900 nM T95286 C1ZL6A 56670360 IC50 = 650 nM T95286 C69SFH 56677195 IC50 = 52000 nM T95286 C9TO7X 56677197 IC50 = 1100 nM T95286 C34CNI 56677199 IC50 = 750 nM T95286 C3QBY9 56677201 IC50 = 300 nM T95286 CS25TR 56680509 IC50 = 300 nM T95286 CKD2Y3 56680511 IC50 = 1200 nM T75596 D08QCJ 5430 IC50 = 44700 nM T75596 D0B1FE 3194 IC50 = 2430 nM T75596 D0KR1N 6918653 EC50 = 0.095 nM T75596 D0KG9M 19910 IC50 = 55 nM T75596 D06WEB 9892113 IC50 = 400 nM T75596 D09OAQ 369976 Ki = 1 nM T75596 CH93VI 2817 IC50 = 55 nM T75596 C1KG9Z 6792 IC50 > 15000 nM T75596 CSU40C 6855 IC50 = 34800 nM T75596 CS0TL4 13224 IC50 = 2030 nM T75596 C9YSM6 125367 IC50 = 0.39 nM T75596 CJW13N 129387 IC50 = 230 nM T75596 CFO0Z8 161167 IC50 = 39800 nM T75596 C41LFG 171397 IC50 = 10400 nM T75596 CMOK67 352929 IC50 = 32900 nM T75596 CVH18S 421108 IC50 = 3810 nM T75596 COPG12 448288 IC50 = 170 nM T75596 C2L7DI 453059 EC50 > 100000 nM T75596 CUQ70N 453063 EC50 > 100000 nM T75596 C7OB8F 461360 IC50 = 41700 nM T75596 CZI5R2 601577 Ki = 6 nM T75596 CB5A1S 612049 IC50 = 24300 nM T75596 C2GEC7 661949 EC50 > 100000 nM T75596 C4TNA0 683337 IC50 = 2660 nM T75596 C62CVW 699784 IC50 = 7680 nM T75596 CULO53 930716 EC50 > 100000 nM T75596 CY4N9Q 935986 EC50 > 100000 nM T75596 C8HIA7 937982 EC50 > 100000 nM T75596 CC4F6Z 1042891 IC50 = 3900 nM T75596 CWNG75 1070711 IC50 = 25800 nM T75596 C5PE1C 1400162 IC50 = 11000 nM T75596 C3AI7O 2725962 IC50 > 100000 nM T75596 CU61SY 2725966 IC50 > 100000 nM T75596 C8Q6VT 2725991 IC50 > 100000 nM T75596 CTS7L9 2725999 IC50 > 100000 nM T75596 CS02AC 2740170 IC50 = 14000 nM T75596 C15MSF 2740173 IC50 = 13000 nM T75596 C6OE0C 2740174 IC50 = 9000 nM T75596 CAHV18 2795593 IC50 > 100000 nM T75596 C9NOS2 2796249 IC50 > 100000 nM T75596 CGI28F 2818423 EC50 > 100000 nM T75596 CIM5V2 3012947 IC50 = 4970 nM T75596 CAIC89 3067566 IC50 = 24300 nM T75596 C9ZAO6 3067567 IC50 = 10900 nM T75596 C9KAP7 3067568 IC50 = 2070 nM T75596 CNA7V9 3067580 IC50 = 10200 nM T75596 C1UJE2 4068684 IC50 > 15000 nM T75596 CCMR86 5326770 IC50 = 30 nM T75596 CN48TU 6102685 IC50 = 4200 nM T75596 CL82TX 6400901 Ki = 4 nM T75596 C3AV5I 6419227 Ki = 18 nM T75596 CIQ4X3 6419341 Ki = 3 nM T75596 CZOJ84 6612277 IC50 = 26700 nM T75596 CNE9Y4 9795779 Ki = 0.04 nM T75596 COMD87 9796214 Ki = 0.07 nM T75596 CO4A3U 9796249 Ki = 5.7 nM T75596 CL75CH 9798133 Ki = 34 nM T75596 C1CR4P 9798321 Ki > 10000 nM T75596 C9XSQ3 9812807 Ki = 41 nM T75596 CAVT12 9812842 Ki = 112 nM T75596 C3EXY0 9814061 Ki = 1 nM T75596 CM5UV3 9814912 Ki = 1 nM T75596 C4UYP5 9815283 Ki = 300 nM T75596 C84KGU 9817701 Ki = 7.762 nM T75596 CJ0K9H 9818391 Ki = 0.43 nM T75596 CC3N7B 9818421 Ki = 4 nM T75596 CQ25OP 9833992 Ki = 260 nM T75596 CFXC18 9839339 Ki = 3.467 nM T75596 C8GXW7 9840569 Ki = 3.3 nM T75596 C0L6OX 9840663 Ki = 0.61 nM T75596 C8M5ZB 9840776 Ki = 4.8 nM T75596 CY1R2C 9861602 Ki = 6.1 nM T75596 CLWJ08 9861819 Ki = 3.1 nM T75596 CQ2GO7 9861976 Ki = 5.2 nM T75596 C98QGX 9862331 Ki = 0.13 nM T75596 CZ78TY 9862362 Ki = 23 nM T75596 C4CAD2 9877457 Ki = 52 nM T75596 C7N9PW 9877511 Ki = 150 nM T75596 C3FC2V 9877859 Ki > 1000 nM T75596 C0CQ9U 9883247 Ki = 0.05 nM T75596 C8EH7L 9883611 Ki = 1.778 nM T75596 C4DC0Q 9884688 Ki = 2.1 nM T75596 C02NYB 9898901 Ki = 337 nM T75596 CCU0I1 9900824 Ki = 0.04 nM T75596 C6T0QK 9904508 Ki = 100 nM T75596 CGZ87A 9905053 Ki = 7.762 nM T75596 CY6I7S 9906523 Ki = 1.5 nM T75596 CKU69T 9920495 Ki = 30 nM T75596 CD8RU5 9920578 Ki > 1000 nM T75596 CL81SX 9922371 IC50 = 600 nM T75596 C4MRZ1 9927000 Ki = 2.5 nM T75596 C4XH9D 9935823 IC50 = 0.96 nM T75596 C0DVR7 9942221 Ki = 3 nM T75596 CERH63 9942963 Ki = 29 nM T75596 C8T5SE 9948612 Ki = 6.5 nM T75596 CUQ39J 9948865 Ki = 1.6 nM T75596 C2PCN3 9964175 Ki = 280 nM T75596 C1YDB5 9964176 Ki = 6 nM T75596 CSRJ64 9964177 Ki = 8 nM T75596 CO52UI 10006629 IC50 = 380 nM T75596 C95BKD 10077016 IC50 = 400 nM T75596 CH3Q7T 10125949 Ki = 24 nM T75596 C6HM5R 10171739 Ki = 1.7 nM T75596 C6VAD2 10171940 Ki = 0.5 nM T75596 CS64TM 10198172 Ki = 1000 nM T75596 CK8AU4 10245616 IC50 = 55 nM T75596 CFU74N 10255531 IC50 = 56 nM T75596 CW4Q9M 10286210 Ki = 0.75 nM T75596 C4LCI9 10286315 Ki = 0.3 nM T75596 CR9K3B 10308455 Ki = 9.1 nM T75596 CMC03E 10425401 Ki = 164000 nM T75596 CFI63J 10650951 IC50 > 50000 nM T75596 C2Q5PA 11120072 IC50 = 53600 nM T75596 CV7C9L 11173284 Ki = 16 nM T75596 C6ET5U 11389807 Ki = 13 nM T75596 CG4FJ6 11496773 IC50 = 190 nM T75596 CMW93D 11503087 IC50 = 270 nM T75596 CVZ6U1 11503191 IC50 = 440 nM T75596 C4I1GC 11503764 IC50 = 20 nM T75596 COGX12 11504270 IC50 = 440 nM T75596 CM6P1N 11506493 Ki = 52 nM T75596 C64JAI 11510709 IC50 = 260 nM T75596 COZ91G 11510858 EC50 = 65 nM T75596 C2MU3R 11510884 IC50 <= 19 nM T75596 C4DTP0 11511194 IC50 = 45 nM T75596 CVTB02 11511667 EC50 = 18000 nM T75596 C7IDU1 11513930 IC50 = 48400 nM T75596 C5TWZ2 11517700 IC50 = 52 nM T75596 C5M4HF 11517890 IC50 = 34.67 nM T75596 CW1N7A 11517913 IC50 = 15 nM T75596 CVQ2C0 11518198 IC50 = 17 nM T75596 C0J8XD 11518243 EC50 = 150 nM T75596 CW48PY 11525062 IC50 = 69 nM T75596 CZ8QH9 11526094 IC50 = 109.65 nM T75596 C2TF7I 11526705 IC50 = 150 nM T75596 C95SUV 11533113 IC50 = 37 nM T75596 C07JIU 11533183 IC50 = 210 nM T75596 CN8IX5 11533642 IC50 = 52 nM T75596 C0X6YF 11535861 IC50 = 40600 nM T75596 C6W1EH 11539389 IC50 = 34.67 nM T75596 C4BFI9 11540018 IC50 = 62 nM T75596 C9VDQ7 11541144 IC50 = 54.95 nM T75596 CBZ89Y 11543088 IC50 = 32900 nM T75596 CF2Y1J 11546119 EC50 = 3000 nM T75596 CD6VJ1 11546431 IC50 = 9 nM T75596 CC79UZ 11546910 IC50 = 5700 nM T75596 CX46VS 11547100 IC50 = 18.2 nM T75596 CIK39Q 11554308 IC50 = 19 nM T75596 CK9TP7 11555354 IC50 = 42 nM T75596 C6RZ4S 11561873 IC50 = 20 nM T75596 CQE7Y4 11561929 IC50 = 150 nM T75596 CNV16Y 11564819 IC50 = 28400 nM T75596 CVP3S4 11568437 IC50 = 12 nM T75596 C6C8XJ 11569061 IC50 = 10 nM T75596 C1SMK8 11569838 IC50 = 170 nM T75596 CS4W8A 11573782 IC50 = 12.88 nM T75596 C6QEW5 11575296 IC50 <= 48 nM T75596 CF9V5T 11575873 EC50 = 110 nM T75596 C47XDB 11576038 IC50 = 52.48 nM T75596 CFTG74 11576103 IC50 = 30 nM T75596 C5C3WZ 11576138 IC50 = 16 nM T75596 CYT7U0 11576158 IC50 = 15 nM T75596 C3OSB1 11576532 IC50 = 43 nM T75596 C9LOY8 11576709 IC50 = 37 nM T75596 CCW7F4 11576736 IC50 = 25 nM T75596 C27GFR 11576769 IC50 = 51 nM T75596 C4S8IK 11577513 EC50 = 460 nM T75596 CDY2H6 11583139 IC50 = 12 nM T75596 CH5CK0 11583415 IC50 = 20 nM T75596 CLE9P8 11583793 EC50 = 360 nM T75596 CH3TJ4 11590100 IC50 = 84 nM T75596 C8PS9W 11597423 IC50 = 17 nM T75596 CUSH60 11597629 IC50 = 30 nM T75596 CA53XH 11597839 IC50 = 17 nM T75596 C1S6QC 11598299 IC50 = 59 nM T75596 C7D4JU 11601120 IC50 = 28000 nM T75596 CM1UG0 11604661 IC50 = 12 nM T75596 CCBE09 11605641 IC50 = 56 nM T75596 CDXW62 11606154 IC50 = 69.18 nM T75596 CT6DL1 11613481 IC50 = 67 nM T75596 CO86NM 11627001 IC50 = 21.88 nM T75596 C1KE5L 11627073 IC50 = 180 nM T75596 C4I2TE 11627706 IC50 = 680 nM T75596 CK4E9Y 11633065 IC50 = 240 nM T75596 C29GWE 11633695 IC50 = 31 nM T75596 C4N9IS 11633910 IC50 = 25 nM T75596 C4ZI7K 11633995 IC50 = 180 nM T75596 CRNL60 11634034 IC50 = 46 nM T75596 CXY74E 11634668 EC50 = 23 nM T75596 CPC84K 11634719 IC50 = 210 nM T75596 CNI6W5 11641405 IC50 = 31 nM T75596 C5RNZ8 11641875 IC50 = 110 nM T75596 CK5AU6 11642511 IC50 = 1400 nM T75596 C42QWY 11644224 IC50 = 38400 nM T75596 CEW1L5 11648539 IC50 = 31 nM T75596 CA6R0P 11648766 EC50 = 270 nM T75596 CVK29M 11649022 EC50 = 1900 nM T75596 C8IAF5 11649266 IC50 = 109.65 nM T75596 CZ2ET7 11651732 IC50 = 44100 nM T75596 CS74DB 11655265 IC50 = 490 nM T75596 C69TBE 11656079 IC50 = 17 nM T75596 C9W5GQ 11662880 IC50 = 66 nM T75596 CEJ83Y 11663131 EC50 = 120 nM T75596 CW2F3C 11663690 IC50 = 690 nM T75596 CJ7V3D 11668537 IC50 = 13 nM T75596 C17VLH 11669769 IC50 = 38 nM T75596 C8QEX6 11670027 IC50 = 11000 nM T75596 CFR4X3 11670580 IC50 = 44 nM T75596 CT9C4Y 11676623 IC50 = 16.98 nM T75596 C07VCQ 11677588 IC50 = 25.7 nM T75596 CRK0X9 11678284 IC50 = 70 nM T75596 C9FZK3 11680001 IC50 = 36400 nM T75596 CIZU85 11683398 EC50 = 110 nM T75596 C8MWD1 11684506 IC50 = 45.71 nM T75596 CD59CW 11684804 IC50 = 77 nM T75596 C3DC5T 11691459 IC50 = 19.05 nM T75596 CHFJ56 11692001 IC50 = 790 nM T75596 C17UFZ 11705233 IC50 = 430 nM T75596 CQT84D 11705551 IC50 = 59 nM T75596 CHXZ40 11713345 EC50 = 510 nM T75596 C73OQV 11719438 IC50 = 3300 nM T75596 CC2OX1 11719751 EC50 = 120 nM T75596 CIT6R8 11720061 IC50 = 26 nM T75596 CN9D1L 11809364 IC50 > 300000 nM T75596 C4BH7P 11822575 IC50 = 8000 nM T75596 CU02JB 13003166 IC50 = 320 nM T75596 C5FJ2G 13650133 IC50 = 935 nM T75596 C82DRK 13673571 IC50 = 5440 nM T75596 C3INS9 13673578 IC50 = 13900 nM T75596 CNU31O 13673587 IC50 = 6790 nM T75596 C0Q3ZD 13673594 IC50 = 3430 nM T75596 C5UY4R 14119495 IC50 = 9130 nM T75596 CBUC49 15516886 IC50 = 5700 nM T75596 CDC80H 15516888 IC50 = 8000 nM T75596 C5I0OT 16005032 IC50 = 2000 nM T75596 CL19UX 16005033 IC50 = 1600 nM T75596 C0QOY1 16005035 IC50 = 1300 nM T75596 CR7H6K 16005036 IC50 = 3800 nM T75596 CRM50J 16005070 IC50 = 700 nM T75596 CWYL26 16005072 IC50 = 1000 nM T75596 C9RB6I 16102135 EC50 = 5.3 nM T75596 CNO01Y 16129576 Ki = 2 nM T75596 CN7MU8 16755845 Ki = 0.9 nM T75596 CG3LP0 16755846 Ki = 21 nM T75596 CUJ2L4 16755847 Ki = 7 nM T75596 CP6B1U 16755848 Ki = 0.7 nM T75596 CQO0T2 16755849 Ki = 135 nM T75596 C7KT3W 16755850 Ki = 10 nM T75596 C1RJM0 16755851 Ki = 0.41 nM T75596 CMO09N 16755952 Ki = 1.3 nM T75596 C3SFJ4 16755953 Ki = 0.9 nM T75596 CWB10M 16755954 Ki = 0.9 nM T75596 C9S0BU 16755955 Ki = 2.7 nM T75596 CZ3IB5 16755956 Ki = 0.5 nM T75596 CEC5Q8 16755957 Ki = 3.8 nM T75596 CU8Y9P 16755958 Ki = 0.8 nM T75596 CV64QT 16756053 Ki = 740 nM T75596 C3JZ6H 16756054 Ki > 2000 nM T75596 CRQ7J0 16756055 Ki > 2000 nM T75596 CL92YI 16756056 Ki = 350 nM T75596 C3AC6K 16756057 Ki > 2000 nM T75596 C5JLQ1 16756058 Ki > 2000 nM T75596 C85OMB 16756059 Ki = 650 nM T75596 C87AFL 16756160 Ki = 480 nM T75596 CM3QS0 16756161 Ki = 1700 nM T75596 C79ZIL 16756162 Ki = 5.7 nM T75596 C0RE6I 16756163 Ki = 3 nM T75596 C6Z0PU 16756164 Ki = 6.5 nM T75596 C9K7EV 16756165 Ki = 1.5 nM T75596 CVO78N 16756166 Ki = 1300 nM T75596 CCA8Y6 16756167 Ki > 10000 nM T75596 CN09YM 16756265 Ki = 15 nM T75596 C0S5LM 16756266 Ki = 66 nM T75596 C3KQN2 16756267 Ki = 1 nM T75596 CR65AJ 16756268 Ki = 3 nM T75596 CH1DV4 16756269 Ki = 24 nM T75596 CN10KR 16757237 Ki = 2.5 nM T75596 CQ4TZ5 16757238 Ki = 61 nM T75596 CT5NZ9 16757239 Ki = 0.23 nM T75596 C4LW6H 16757240 Ki = 2.4 nM T75596 C2KJD4 16757241 Ki = 3.7 nM T75596 CYF2H7 16757242 Ki = 3.3 nM T75596 CHI8J9 16757243 Ki = 0.15 nM T75596 C6G3MI 16757244 Ki = 3.8 nM T75596 CLX71H 16757340 Ki = 3.6 nM T75596 CWIO01 16757341 Ki > 10000 nM T75596 C5QSH8 16757342 Ki = 0.65 nM T75596 CZ1FI4 16757343 Ki = 1.2 nM T75596 CZ65WX 16757344 Ki = 5.2 nM T75596 C1LKY5 16757345 Ki = 0.52 nM T75596 CG35HL 16757346 Ki = 18 nM T75596 CAYS87 16757347 Ki = 0.16 nM T75596 CUJ8E9 16757446 Ki = 1.7 nM T75596 C1O0RW 16757447 Ki = 18 nM T75596 C43EZH 16757448 Ki > 1000 nM T75596 CP7U2O 16757449 Ki = 1.3 nM T75596 CO74PX 16757450 Ki = 4 nM T75596 CWHZ37 16757451 Ki = 9.6 nM T75596 CP18LO 16757452 Ki = 8.3 nM T75596 CX24TA 17748229 IC50 = 87 nM T75596 C4DV3T 20660272 IC50 = 1300 nM T75596 CM9PK0 21455599 IC50 = 50.12 nM T75596 CY89WP 23644716 IC50 = 4200 nM T75596 C2A4SZ 23647744 IC50 = 16 nM T75596 CE30PG 23647749 IC50 = 55 nM T75596 CYO2D5 23647750 IC50 = 510 nM T75596 C4YUS0 23647754 IC50 = 50 nM T75596 CH89QX 23647755 IC50 = 190 nM T75596 CD6Q5V 23647756 IC50 = 270 nM T75596 CCN67D 23647757 IC50 = 130 nM T75596 CQ39MH 23647759 IC50 = 20 nM T75596 CQBI56 23647760 IC50 = 2600 nM T75596 CSQ0R7 23647761 IC50 = 27 nM T75596 CD53RS 23647762 IC50 = 60 nM T75596 C4SAZ0 23647763 IC50 = 16 nM T75596 CX2H4C 23647764 IC50 = 150 nM T75596 CN70TP 23647765 IC50 = 1300 nM T75596 C9YW1V 23647766 IC50 = 8000 nM T75596 CCF62S 23647767 IC50 = 2500 nM T75596 CC63AD 23647768 IC50 = 11 nM T75596 CVG9D6 23647769 IC50 = 8 nM T75596 C8OPE9 23647770 IC50 = 20 nM T75596 CJD75W 23647771 IC50 = 1000 nM T75596 CH0US8 23647772 IC50 = 36000 nM T75596 C3YWX9 23647773 IC50 = 14000 nM T75596 C7RGV3 23647774 IC50 = 15 nM T75596 C5TD7R 23647775 IC50 = 38 nM T75596 C54DMX 23647776 IC50 = 46 nM T75596 CT5DX3 23647777 IC50 = 5800 nM T75596 C1XHP4 23647778 IC50 = 230 nM T75596 CE8AU6 23647779 IC50 = 555 nM T75596 C8P1VI 23647780 IC50 = 85 nM T75596 CH87IP 23647781 IC50 = 10 nM T75596 CU36YX 23647782 IC50 = 18 nM T75596 C7M9NT 23647783 IC50 = 85 nM T75596 CFHV96 23647784 IC50 = 26 nM T75596 C3CGL0 23647785 IC50 = 96 nM T75596 C42CVJ 24728213 IC50 = 2800 nM T75596 C0UG6Z 44337882 IC50 = 755 nM T75596 CTB9K0 44337913 IC50 = 230 nM T75596 CUX7V9 44337914 IC50 = 158 nM T75596 C0O6KM 44337931 IC50 = 45 nM T75596 C6VS3E 44337932 IC50 = 58 nM T75596 C85SAJ 44337936 IC50 = 177 nM T75596 CSIO36 44337940 IC50 = 82 nM T75596 C4SQ2Z 44337959 IC50 = 217 nM T75596 CM5DN8 44337963 IC50 = 2200 nM T75596 C6FN9K 44337998 IC50 = 98 nM T75596 CWY3K6 44337999 IC50 = 33 nM T75596 CZ3K4H 44338000 IC50 = 46 nM T75596 CLT61H 44338001 IC50 = 35 nM T75596 C1WPH0 44338006 IC50 = 209 nM T75596 C17CVQ 44338007 IC50 = 169 nM T75596 CK98CU 44338009 IC50 = 100 nM T75596 CVB4O3 44338054 IC50 = 308 nM T75596 C9HWD2 44338069 IC50 = 356 nM T75596 CML7D1 44338070 IC50 = 67 nM T75596 CA69UZ 44338268 IC50 = 43 nM T75596 C70ABO 44343208 IC50 = 8000 nM T75596 C2P9OQ 44378659 Ki = 1300000 nM T75596 CLRN70 44378660 Ki = 91000 nM T75596 C9DC4A 44378725 Ki = 600000 nM T75596 CRD8O0 44381636 IC50 = 160 nM T75596 C6E3UH 44381637 IC50 = 16000 nM T75596 CZ6RG7 44381638 IC50 = 900 nM T75596 CSQ0W5 44381639 IC50 = 1000 nM T75596 C70VGJ 44381640 IC50 = 460 nM T75596 CSP60T 44381644 IC50 = 35000 nM T75596 CR7J1I 44381648 IC50 = 310 nM T75596 CXW14E 44381649 IC50 = 460 nM T75596 CP84UL 44381661 IC50 = 14000 nM T75596 CGC5S6 44381662 IC50 = 4300 nM T75596 CCY8A4 44381663 IC50 = 12500 nM T75596 CD6T8L 44381665 IC50 = 1100 nM T75596 CA27TF 44381668 IC50 = 120 nM T75596 CNJ74O 44381669 IC50 = 140 nM T75596 C1UIR6 44381689 IC50 = 590 nM T75596 CE82LP 44381690 IC50 = 970 nM T75596 CV65EN 44381693 IC50 = 3600 nM T75596 C2UKS5 44381700 IC50 = 70 nM T75596 CZM56N 44381703 IC50 = 8600 nM T75596 CAMB80 44381704 IC50 = 5300 nM T75596 C0IU7J 44381705 IC50 = 2400 nM T75596 C0S9NU 44381720 IC50 = 20 nM T75596 C0TI6L 44381731 IC50 = 1200 nM T75596 C46EFV 44381733 IC50 = 1800 nM T75596 CLA25E 44381734 IC50 = 1600 nM T75596 CX7KI3 44381742 IC50 = 130 nM T75596 CL0KD5 44381743 IC50 = 50 nM T75596 CC1PK9 44381755 IC50 = 50 nM T75596 C4PTD7 44381756 IC50 = 480 nM T75596 C5GTW7 44381764 IC50 = 320 nM T75596 C4SNP1 44381771 IC50 = 60 nM T75596 C9YH2Q 44381772 IC50 = 270 nM T75596 C1XCO0 44381773 IC50 = 290 nM T75596 CO60XF 44381796 IC50 = 1500 nM T75596 C9WBI4 44381812 IC50 = 200 nM T75596 CPQK86 44381823 IC50 = 1400 nM T75596 CZR3U0 44381824 IC50 = 290 nM T75596 CG8F0L 44381857 IC50 > 100000 nM T75596 CKS79L 44381893 IC50 = 74000 nM T75596 CB09OX 44381894 IC50 = 51000 nM T75596 C5APZ6 44381897 IC50 = 250 nM T75596 C1BCZ9 44381901 IC50 = 1100 nM T75596 CUP5A0 44381903 IC50 = 3500 nM T75596 CW3I2S 44381904 IC50 = 2600 nM T75596 CA2F3C 44381909 IC50 = 40 nM T75596 CEW7Z9 44381912 IC50 = 1600 nM T75596 CNMH89 44381916 IC50 = 600 nM T75596 CSB3V8 44381933 IC50 = 120 nM T75596 CQR38H 44381935 IC50 = 620 nM T75596 CAHN94 44381940 IC50 = 2700 nM T75596 CAXC40 44381941 IC50 = 420 nM T75596 CNE58C 44381946 IC50 = 30 nM T75596 CH2KV7 44381952 IC50 = 1000 nM T75596 C91HWB 44381954 IC50 = 500 nM T75596 C63FRA 44381955 IC50 = 190 nM T75596 CT5GL2 44381961 IC50 = 50 nM T75596 C0KYX6 44381962 IC50 = 1700 nM T75596 CK7N0V 44381963 IC50 = 50 nM T75596 CF20MK 44381969 IC50 = 4100 nM T75596 C12GXS 44381973 IC50 = 210 nM T75596 CC9I0D 44381976 IC50 = 850 nM T75596 C68WOA 44381980 IC50 = 6100 nM T75596 CCH82P 44381981 IC50 = 1500 nM T75596 C8JEP3 44381987 IC50 = 20 nM T75596 C7MHO1 44381988 IC50 = 560 nM T75596 CF60YV 44381993 IC50 = 1200 nM T75596 CZX82N 44381997 IC50 = 50 nM T75596 CO18AS 44381998 IC50 = 50 nM T75596 CDX0N9 44381999 IC50 = 430 nM T75596 C8ZS3M 44382016 IC50 = 51000 nM T75596 C9NE3W 44382027 IC50 = 140 nM T75596 CGS36C 44382028 IC50 = 120 nM T75596 CRW8B3 44382049 IC50 = 4900 nM T75596 CA3OQ9 44382050 IC50 = 3200 nM T75596 CJR46W 44382074 IC50 = 240 nM T75596 C7WK8D 44382075 IC50 = 14000 nM T75596 CC42PH 44382076 IC50 = 1600 nM T75596 CR3TX2 44382078 IC50 = 830 nM T75596 CNMF84 44382132 IC50 = 250 nM T75596 CD63HL 44382395 IC50 = 800 nM T75596 C7HA9B 44382396 IC50 = 500 nM T75596 CF2Y5T 44382446 IC50 = 1100 nM T75596 C6ZPD8 44382483 IC50 = 310 nM T75596 C0OZ1L 44382517 IC50 = 700 nM T75596 CHEX78 44382518 IC50 = 2100 nM T75596 C5A7XT 44382564 IC50 = 1300 nM T75596 C18GSZ 44382565 IC50 = 42000 nM T75596 C1UE5V 44382789 IC50 = 900 nM T75596 C9I2CT 44383748 IC50 = 1.2 nM T75596 CNC81X 44383750 IC50 = 0.8 nM T75596 CVK95D 44383841 IC50 = 1.2 nM T75596 CNO72W 44384130 IC50 = 8.9 nM T75596 CK5Q2E 44385026 IC50 = 1.7 nM T75596 CVQL03 44385027 IC50 = 0.51 nM T75596 C38FTJ 44385040 IC50 = 0.43 nM T75596 CS7ZL5 44413082 IC50 <= 18 nM T75596 CK9G3B 44413210 IC50 = 15 nM T75596 CUL1R4 44415938 IC50 = 33800 nM T75596 CAZ5D9 44416035 IC50 = 57500 nM T75596 C0EYD9 44416055 IC50 = 13200 nM T75596 CJ1UH7 44416119 IC50 = 3230 nM T75596 C1QC5U 44553054 IC50 = 2200 nM T75596 CRQ5T3 44553055 IC50 = 8600 nM T75596 C9D6AC 44553226 IC50 = 450 nM T75596 CGF8P5 44553573 IC50 = 2800 nM T75596 C48OCV 44553900 IC50 > 50000 nM T75596 C3U5VD 44554434 IC50 = 230 nM T75596 C83QND 44590979 IC50 > 100000 nM T75596 C5WP7Y 44720028 IC50 = 9 nM T75596 CU32GN 45267083 IC50 > 50000 nM T75596 CS6KU9 46842838 IC50 = 110 nM T75596 CHL9S5 46865372 IC50 = 560 nM T75596 CKX7D0 52942444 IC50 = 91.2 nM T75596 C3AI8T 52943911 IC50 = 128.82 nM T75596 CL1VK9 52946375 IC50 = 52.48 nM T75596 CLM52E 54754514 IC50 = 930 nM T75596 CX4A7W 56563890 IC50 > 100000 nM T75596 C6MHX1 56659884 IC50 = 1920 nM T75596 CI5U1C 56663343 IC50 = 30710 nM T75596 CWD19S 56663344 IC50 = 5910 nM T75596 C12DLZ 56666768 IC50 = 7290 nM T75596 CYR14U 56666774 IC50 = 11780 nM T75596 C0YI1P 56666776 IC50 = 3450 nM T75596 CN3MW5 56670208 IC50 = 1840 nM T75596 CL5BD1 56670209 IC50 = 3950 nM T75596 C8FT5G 56673730 IC50 = 5370 nM T75596 CG5J6H 56677036 IC50 = 6010 nM T75596 CGH0O5 56677037 IC50 = 12390 nM T75596 CJ3HB6 56680364 IC50 = 4800 nM T75596 C43ZPV 56683700 IC50 = 17660 nM T75596 C0PB7Y 56683701 IC50 = 2240 nM T75596 C92SHF 56959518 IC50 = 220 nM T75596 C1INR0 56959669 IC50 = 240 nM T75596 CJX9B2 56959670 IC50 = 140 nM T75596 C3A4EP 56959817 IC50 = 440 nM T75596 C5S3AD 56959819 IC50 = 140 nM T75596 C9Y6XF 56959820 IC50 = 50 nM T75596 C2LVY4 56960117 IC50 = 380 nM T75596 CLRM47 56960253 IC50 = 170 nM T75596 C0HOV4 56960254 IC50 = 57 nM T75596 CAX3V7 56960533 IC50 = 410 nM T75596 CC3GI2 56960810 IC50 = 740 nM T75596 C0KQ2X 56960811 IC50 = 480 nM T75596 C0MKX4 56960816 IC50 = 80 nM T75596 CI19KQ 56960946 IC50 = 60 nM T75596 CQ7T2M 56960952 IC50 = 700 nM T75596 COU9T2 58279815 IC50 > 100000 nM T75596 CB31IC 58279829 IC50 > 100000 nM T75596 CJUP62 60043945 EC50 = 6.5 nM T75596 CBY8K5 66995905 IC50 = 1800 nM T75596 CET5F2 67315720 IC50 > 50000 nM T75596 C2M9SU 68347001 EC50 > 300000 nM T75596 CI1J8B 68347004 EC50 > 300000 nM T75596 C7VK9T 68347007 IC50 = 22000 nM T75596 C6S0MJ 68347012 IC50 = 114000 nM T75596 CR60HY 68347026 IC50 > 300000 nM T75596 CF7A0K 68347055 IC50 = 188000 nM T75596 C4I5BQ 68347057 EC50 = 53000 nM T75596 CFKS17 68347135 IC50 = 9400 nM T75596 C7HS6V 68347136 IC50 = 62000 nM T75596 CT5W9F 68347138 IC50 = 108000 nM T75596 COS5C6 68347139 IC50 = 197000 nM T75596 CZRK60 68347140 IC50 = 95000 nM T75596 CT19PO 68347143 IC50 = 101000 nM T75596 C2Y0IB 68347313 IC50 > 300000 nM T75596 C26ZEC 68347339 EC50 > 300000 nM T75596 CWDR01 70683062 IC50 = 57 nM T75596 C0JNV4 70689368 IC50 = 25 nM T75596 CLG35E 71472495 IC50 < 50 nM T75596 CL8H2B 71602394 EC50 = 14000 nM T75596 C5TPO1 71602459 EC50 = 1100 nM T75596 C5LCD8 71602460 EC50 = 28000 nM T75596 CCB58N 71602527 EC50 > 30000 nM T75596 CMWJ83 71602528 EC50 > 30000 nM T75596 CKBD52 71602529 EC50 > 30000 nM T75596 CDKF42 71602530 EC50 = 31000 nM T75596 C31MVT 71602531 EC50 > 100000 nM T75596 CC78SK 71602588 EC50 > 30000 nM T75596 C7CT2W 71602589 EC50 > 300000 nM T75596 C61ABC 71602590 EC50 > 100000 nM T75596 CXCQ63 71602591 EC50 > 100000 nM T75596 CBN17L 71602592 EC50 > 30000 nM T75596 C7WA2F 71602646 EC50 > 300000 nM T75596 CVG89D 71602647 EC50 = 16000 nM T75596 CC2R3T 71602648 EC50 > 300000 nM T75596 CP60LJ 71602649 EC50 > 300000 nM T75596 C5UP7K 71602650 EC50 > 300000 nM T75596 C1UV4S 71602693 EC50 > 300000 nM T75596 CGTV32 71602694 EC50 > 300000 nM T75596 CV5XT2 71602695 EC50 > 100000 nM T75596 CY5S8M 71602696 EC50 > 200000 nM T75596 C5ZGU1 71602697 EC50 > 200000 nM T75596 C0WOA4 71602745 EC50 > 200000 nM T75596 CM2VE7 71602796 EC50 > 200000 nM T75596 CQ6Y1W 71603176 EC50 > 30000 nM T75596 CY60QJ 71603177 EC50 > 30000 nM T75596 COE76Q 71603178 EC50 > 300000 nM T75596 CZM7C8 71603179 EC50 > 300000 nM T75596 C20ZQI 71603235 EC50 = 1200 nM T75596 CSF38G 71603236 EC50 = 1200 nM T75596 CLXH32 71603237 EC50 = 14000 nM T75596 CV5Q1A 71603238 EC50 = 1700 nM T75596 C2P5FS 71614682 IC50 = 2080 nM T75596 CUP3N9 71614683 IC50 = 4790 nM T75596 C1CG2M 71614684 IC50 = 6330 nM T75596 C6WK7Y 71614685 IC50 = 10040 nM T75596 C4QB8A 71614878 IC50 = 7920 nM T75596 C8WTV4 71614879 IC50 = 8410 nM T75596 C9RPO3 71614880 IC50 = 10710 nM T75596 CE9X6T 71614881 IC50 = 12660 nM T75596 C4T9DU 71615081 IC50 = 22030 nM T75596 C92QPX 71615082 IC50 = 18240 nM T75596 C0FTC2 71615083 IC50 = 13950 nM T75596 C5A9GT 71735205 IC50 = 20 nM T75596 CZ3BR1 71735206 IC50 = 11 nM T75596 CGNL45 71735207 IC50 = 4 nM T75596 CS06UR 71735209 IC50 = 3 nM T75596 C1MK3N 71735210 IC50 = 6 nM T75596 CO4L2A 71735375 IC50 = 9 nM T75596 CE0GO2 71815258 IC50 = 94 nM T75596 CCF61D 71815827 IC50 = 62 nM T75596 CSLT73 71815970 IC50 = 160 nM T75596 CE8A4J 71816100 IC50 = 44 nM T75596 CLG1E3 73345794 EC50 > 100000 nM T75596 C2WP7O 73345795 EC50 > 100000 nM T75596 CNKZ64 73345796 EC50 > 100000 nM T75596 CCUG98 73345797 EC50 > 100000 nM T75596 C0C8JI 73345798 EC50 > 100000 nM T75596 C64ZSF 73347280 EC50 > 100000 nM T75596 CN90YL 73347281 EC50 > 100000 nM T75596 C1EV2G 73347282 EC50 > 200000 nM T75596 CH0IL4 73348796 EC50 > 100000 nM T75596 CUH1J4 73348797 EC50 > 100000 nM T75596 CU20ZW 73350374 EC50 > 100000 nM T75596 CG2K3V 73351884 EC50 > 200000 nM T75596 C4N9JC 73353354 EC50 > 100000 nM T75596 CT41OK 73353355 EC50 > 300000 nM T75596 CAK6B5 73353356 EC50 > 100000 nM T75596 C5B3JW 73356423 EC50 > 100000 nM T75596 CN58LK 73356424 EC50 > 100000 nM T75596 C2FV6Y 73425712 EC50 = 251.19 nM T75596 CD5JG2 73426249 IC50 = 12.59 nM T75596 C5P7VZ 73426250 IC50 = 7.943 nM T75596 C48TXH 73426341 IC50 = 5.012 nM T75596 CJ0QN7 73426346 EC50 = 25.12 nM T75596 CM5X1V 73426735 IC50 = 6.31 nM T75596 C4V8EW 73426736 EC50 = 19.95 nM T75596 C48ACZ 88621253 IC50 = 121 nM T75596 C3YCM9 88621311 IC50 = 9980 nM T75596 CEF6R1 89443960 IC50 = 5500 nM T75596 C46EZY 89782850 EC50 = 37 nM T75596 CWH3V4 89783047 IC50 = 10 nM T75596 CAN93M 89783069 IC50 = 21 nM T75596 C1SHB3 89783092 IC50 = 11 nM T75596 C4LV1B 89783137 IC50 = 8 nM T75596 CBH3O6 89783177 IC50 = 8 nM T75596 C72EQS 89783285 IC50 = 8 nM T75596 C3LY2B 89783293 IC50 = 5 nM T75596 C6DE5I 89783377 IC50 = 15 nM T75596 C9RQ3O 89783586 IC50 = 4 nM T75596 CU6B2I 89794927 EC50 = 15 nM T75596 COT8P7 89855771 IC50 = 120 nM T75596 C7HP6U 89855775 IC50 = 52 nM T75596 CY7DH8 89855776 Ki = 4.33 nM T75596 CJN31S 89855779 IC50 = 110 nM T75596 C84GQR 89855793 IC50 = 14 nM T75596 CC2EV5 89855828 IC50 = 30 nM T75596 CJ7G3L 89855860 IC50 = 100 nM T75596 C17GAX 89855873 IC50 = 95 nM T75596 C3Z4IC 89855890 IC50 = 50 nM T75596 C32LKW 89855916 IC50 = 53 nM T75596 CQ63GB 89855918 IC50 = 16 nM T75596 C72SHX 89855938 IC50 = 110 nM T75596 CK67TU 89855943 IC50 = 52 nM T75596 CGU58D 89855953 Ki = 3.36 nM T75596 CK0EX5 89893205 IC50 = 17000 nM T75596 CY12WJ 89893217 IC50 = 550 nM T75596 C57OLX 89893263 IC50 = 860 nM T75596 CW07KQ 89893264 IC50 = 130 nM T75596 CLZ5N7 89893271 IC50 = 90 nM T75596 C3AIE6 89893272 IC50 = 60 nM T75596 CC48DY 89893284 IC50 = 270 nM T75596 C8ZX7O 89893288 IC50 = 280 nM T75596 C0G3IH 89893318 IC50 = 5300 nM T75596 C7F2UR 89893622 Ki = 0.16 nM T75596 CCN1E5 89893636 IC50 = 79 nM T75596 C98JCD 89893658 IC50 = 60 nM T75596 C0GLT6 89893669 IC50 = 90 nM T75596 CE3NI5 89893683 IC50 = 46 nM T75596 C2QOM5 89893711 IC50 = 60 nM T75596 C5M1KL 89893722 IC50 = 90 nM T75596 CEQ2P8 89893732 IC50 = 540 nM T75596 C6GOP2 89893744 IC50 = 12 nM T75596 CF2V1L 89893761 IC50 = 80 nM T75596 CX23BK 90082686 IC50 = 220 nM T75596 CCI08S 98126253 IC50 = 200 nM T75596 C7I4LF 102261763 IC50 = 7570 nM T75596 CP37LV 117832568 IC50 = 9 nM T75596 C23ZUP 118753274 EC50 = 8.8 nM T75596 CPGJ59 118753275 EC50 = 11.7 nM T75596 CU7NP9 118753315 EC50 = 7.1 nM T75596 CVZJ40 118753355 EC50 = 0.3 nM T75596 CE51NI 118753356 EC50 = 1.3 nM T75596 CE3PN1 118870023 IC50 = 72 nM T75596 CVD8B4 118884324 IC50 = 13 nM T75596 C3W2JQ 118917376 IC50 > 100000 nM T75596 C1XZS7 124185467 IC50 = 590 nM T75596 CQO07L 127046305 IC50 = 960 nM T75596 CKB3P7 127046306 IC50 = 220 nM T75596 CJSH70 127046307 IC50 = 730 nM T75596 C9EUK1 127046308 IC50 = 62 nM T75596 C8T4GP 127046309 IC50 = 91 nM T75596 C1H6OK 127046586 IC50 = 360 nM T75596 CR9M3E 127046692 IC50 = 6 nM T75596 CHE2B0 127047126 IC50 = 24000 nM T75596 CT1Z3C 127047212 IC50 = 550 nM T75596 C10DGM 127047414 EC50 = 65 nM T75596 C08NVU 127047863 IC50 = 79 nM T75596 CDIZ79 127047981 IC50 = 5 nM T75596 CC3YA4 127048005 IC50 = 5.012 nM T75596 CBJ84R 127048091 EC50 = 31.62 nM T75596 CXP15S 130307835 IC50 = 200 nM T75596 CNGV45 130307851 Ki = 0.9 nM T75596 CCB1X6 134135510 IC50 = 4470 nM T75596 CP6QB3 134137117 IC50 = 2350 nM T75596 C42XSV 134137805 IC50 = 920 nM T75596 C2WQ6Z 134138481 IC50 = 119200 nM T75596 CP7U3L 134139056 IC50 = 1350 nM T75596 CC1Y6U 134142920 IC50 = 2670 nM T75596 C4IUX3 134143100 IC50 = 6270 nM T75596 C4SA6I 134146877 IC50 = 8850 nM T75596 CK64BT 135446116 Ki > 1000 nM T75596 CGEO38 136442281 IC50 = 1000 nM T75596 C21ETJ 137210068 IC50 = 79.43 nM T75596 CMJ48Z 137636803 IC50 = 38 nM T75596 CB8M5D 137638869 IC50 > 50000 nM T75596 CH7Q2K 155530368 IC50 = 80 nM T75596 D00MUJ 10018850 IC50 = 1100 nM T75596 D02ADV 594397 Ki = 4.2 nM T75596 D02APY 448285 IC50 = 110 nM T75596 D02OAB 761929 IC50 = 37000 nM T75596 D04KUP 17842471 IC50 = 1100 nM T75596 D04MIY 186763 IC50 = 18100 nM T75596 D04SLM 10957430 IC50 = 0.4 nM T75596 D05DCQ 9838682 Ki = 0.5 nM T75596 D07CWJ 6102684 IC50 = 1000 nM T75596 D07PXR 11665659 IC50 = 14900 nM T75596 D08AXA 947740 IC50 = 8000 nM T75596 D08CFL 6917655 IC50 = 0.63 nM T75596 D09KTF 10246233 IC50 = 10000 nM T75596 D0B1LR 134912 IC50 = 10100 nM T75596 D0C0UB 345772 IC50 = 7700 nM T75596 D0FO2B 1923 IC50 = 5600 nM T75596 D0I6RL 11723962 IC50 = 19 nM T75596 D0K5UM 23647758 IC50 = 350 nM T75596 D0K7PS 1069140 IC50 = 9100 nM T75596 D0L4YF 70821 IC50 = 13300 nM T75596 D0L6ZY 542828 IC50 = 9300 nM T75596 D0O3IE 137153 Ki = 70 nM T75596 D0R4KE 10427648 IC50 = 15 nM T75596 D0S5GM 10402833 IC50 = 90 nM T75596 D0UV8T 9942176 Ki > 1000 nM T57392 D00FGR 3599 IC50 > 100000 nM T57392 D00JVR 2267 IC50 = 1000 nM T57392 D00KHM 16362 IC50 > 30000 nM T57392 D00KVO 2082 IC50 > 30000 nM T57392 D00UVA 11556711 IC50 > 10000 nM T57392 D00YZD 54726191 IC50 > 100000 nM T57392 D01AXB 60835 IC50 = 1600 nM T57392 D01JGV 441975 Ki = 3.3 nM T57392 D01ZII 2726 IC50 = 1490 nM T57392 D02DPA 2756 Ki = 77000 nM T57392 D02HED 4748 IC50 = 120 nM T57392 D02VJP 25151504 IC50 = 9200 nM T57392 D03BLF 31307 IC50 > 50000 nM T57392 D03DDR 3034034 IC50 = 10 nM T57392 D03DIG 5284371 IC50 = 104000 nM T57392 D03HFG 5324346 Ki = 8000 nM T57392 D03ROX 2369 IC50 = 66000 nM T57392 D03WEX 9966051 IC50 = 9800 nM T57392 D04CRN 54841 IC50 = 2000 nM T57392 D04JEE 4946 IC50 = 1900 nM T57392 D04NQI 2165 IC50 = 640 nM T57392 D04OSE 4485 IC50 > 50000 nM T57392 D04WFD 4543 IC50 = 2300 nM T57392 D04XGT 31593 IC50 = 77800 nM T57392 D05CEU 941361 IC50 = 7890 nM T57392 D05EAM 4735 IC50 = 10000 nM T57392 D05LBU 5472 IC50 = 4800 nM T57392 D05UVD 33624 IC50 = 11000 nM T57392 D06ABF 3957 IC50 < 100 nM T57392 D06GDY 43815 IC50 = 960 nM T57392 D06GKN 2099 IC50 < 10000 nM T57392 D06MAJ 65906 Ki > 20000 nM T57392 D07ACT 5479530 IC50 > 50000 nM T57392 D07ESC 11561674 IC50 > 10000 nM T57392 D07KSG 2733526 IC50 = 13700 nM T57392 D07UYO 441401 IC50 > 20000 nM T57392 D08VYV 4168 Ki = 960 nM T57392 D09GOS 2812 IC50 = 883 nM T57392 D09IPV 28417 IC50 = 2740 nM T57392 D09OBB 5360696 IC50 = 1800 nM T57392 D09SGV 25154714 IC50 > 100000 nM T57392 D0B4IF 456201 IC50 = 10 nM T57392 D0C3SW 53465279 IC50 = 92100 nM T57392 D0D1AL 3559 IC50 = 3640 nM T57392 D0D4YZ 45375808 IC50 > 100000 nM T57392 D0D9FV 4601 IC50 > 30000 nM T57392 D0EG1I 9926791 IC50 > 52000 nM T57392 D0F9BY 166548 IC50 > 17500 nM T57392 D0G4KG 3828 IC50 > 10000 nM T57392 D0G9YH 2179 Ki = 7500 nM T57392 D0H0KB 5070 IC50 > 25000 nM T57392 D0H0ND 54454 IC50 > 30000 nM T57392 D0H4JM 8969 IC50 = 8.4 nM T57392 D0I1FQ 54671008 IC50 > 50000 nM T57392 D0I2MK 4171 IC50 = 24000 nM T57392 D0K0TC 68617 IC50 = 1400 nM T57392 D0K8KX 5280343 IC50 = 18800 nM T57392 D0K9MY 11243969 IC50 > 50000 nM T57392 D0L0MK 7014 IC50 = 60000 nM T57392 D0MP5H 2966 IC50 = 23800 nM T57392 D0N6RF 65999 IC50 > 50000 nM T57392 D0NJ5H 11450633 IC50 < 10000 nM T57392 D0O3OS 104850 IC50 > 20 nM T57392 D0Q2PE 4539 IC50 > 50000 nM T57392 D0QV5T 54680692 IC50 = 528000 nM T57392 D0R0FE 2520 IC50 > 30000 nM T57392 D0R3JB 4212 IC50 = 76300 nM T57392 D0S5LO 25166913 IC50 > 30000 nM T57392 D0T0KA 4474 IC50 = 1590 nM T57392 D0T6WN 6451164 IC50 = 3410 nM T57392 D0T8XB 44513473 IC50 > 10000 nM T57392 D0V7CF 5362440 IC50 > 30000 nM T57392 D0V8QT 2708 IC50 = 65100 nM T57392 D0W7WC 16220172 IC50 > 20000 nM T57392 D0Y4JJ 2351 IC50 > 30000 nM T57392 D0Y7LD 222284 IC50 > 100000 nM T57392 D0Z1RV 135398737 IC50 = 18000 nM T57392 D0Z3DY 2333 IC50 > 50000 nM T57392 D0Z7KE 3784 IC50 = 4790 nM T57392 D0ZU9R 392622 IC50 = 2300 nM T57392 D00DRL 44137946 IC50 > 100000 nM T57392 D00JFE 56941241 IC50 > 20000 nM T57392 D00RYA 16750271 IC50 > 10000 nM T57392 D01DDN 56950369 IC50 > 50000 nM T57392 D01LCC 17754438 IC50 > 30000 nM T57392 D02AAO 10368812 IC50 > 10000 nM T57392 D02AIN 122678117 IC50 > 20000 nM T57392 D02EEJ 6479267 IC50 > 100000 nM T57392 D02NNV 3038525 IC50 > 40000 nM T57392 D02QWY 24785538 IC50 > 40000 nM T57392 D03AJU 44139752 IC50 > 10000 nM T57392 D03FOP 68947304 IC50 > 27000 nM T57392 D03GNI 2166 IC50 = 7000 nM T57392 D03ISJ 135564632 IC50 > 50000 nM T57392 D03LWG 53235510 IC50 > 10000 nM T57392 D03MZJ 51045 IC50 = 50 nM T57392 D03QHC 49856296 IC50 > 6000 nM T57392 D03SQT 68234908 IC50 > 100000 nM T57392 D03WNG 73051463 IC50 = 9000 nM T57392 D04JTX 66561902 IC50 > 30000 nM T57392 D04MXN 56846693 IC50 > 10000 nM T57392 D04TNT 46851313 IC50 > 10000 nM T57392 D04WUA 219101 IC50 = 4250 nM T57392 D05LRD 59286554 IC50 > 30000 nM T57392 D05OMT 45142457 IC50 = 46170 nM T57392 D05PZB 135398495 IC50 > 10000 nM T57392 D05UYQ 15984937 IC50 = 34000 nM T57392 D06EPO 11192346 IC50 > 30000 nM T57392 D06MHZ 66558287 IC50 = 2200 nM T57392 D06TKI 49857317 IC50 > 50000 nM T57392 D06TQR 76287260 IC50 = 82000 nM T57392 D06ZEO 54674461 IC50 > 50000 nM T57392 D07BXE 71750 IC50 = 48000 nM T57392 D07HZG 11516136 IC50 > 30000 nM T57392 D07OFM 46943432 IC50 >= 33000 nM T57392 D07TEP 10117987 IC50 > 40000 nM T57392 D08AOZ 86582336 IC50 > 40000 nM T57392 D08PMW 9951995 IC50 = 35000 nM T57392 D08SCL 46190695 IC50 > 50000 nM T57392 D08UGX 60652 IC50 = 4760 nM T57392 D08VSQ 59336911 IC50 > 40000 nM T57392 D09DXX 71571306 IC50 > 100000 nM T57392 D09RII 71602803 IC50 = 148000 nM T57392 D09WYL 11634973 IC50 > 100000 nM T57392 D0A7ZK 56944144 IC50 > 20000 nM T57392 D0B5HF 44476893 IC50 > 50000 nM T57392 D0BM7M 11488320 IC50 > 10000 nM T57392 D0C8DD 11552706 IC50 >= 79432.82 nM T57392 D0C9PZ 91754484 IC50 > 50000 nM T57392 D0CB2B 23653789 IC50 = 35000 nM T57392 D0CG8S 71305058 IC50 > 25000 nM T57392 D0CW8S 71657619 IC50 = 6500 nM T57392 D0DH5X 44472635 IC50 > 100000 nM T57392 D0E0JO 117857370 EC50 > 100000 nM T57392 D0EB5N 25185057 IC50 > 25000 nM T57392 D0EM4S 17751090 IC50 > 25000 nM T57392 D0EY0A 42636350 IC50 > 30000 nM T57392 D0F4JK 11547499 IC50 > 30000 nM T57392 D0F4ZY 5311037 IC50 > 40000 nM T57392 D0F5NJ 1615 Ki = 12900 nM T57392 D0F6YM 3035000 IC50 > 50000 nM T57392 D0FD6D 11751922 IC50 > 30000 nM T57392 D0G5XV 135565884 IC50 > 30000 nM T57392 D0G7UX 5284373 IC50 > 100000 nM T57392 D0G9AW 59473233 IC50 > 10000 nM T57392 D0GC5H 123879 IC50 > 30000 nM T57392 D0H8OA 46917559 IC50 = 11000 nM T57392 D0H9DA 54761306 IC50 > 10000 nM T57392 D0H9SX 6914657 IC50 > 10000 nM T57392 D0HR7P 50515 IC50 = 39600 nM T57392 D0HS5V 11234052 IC50 > 40000 nM T57392 D0I2XM 3038500 IC50 = 11000 nM T57392 D0I3LO 91933883 IC50 > 20000 nM T57392 D0I3TU 45268455 IC50 > 30000 nM T57392 D0I4PW 60164925 IC50 > 50000 nM T57392 D0I8FV 5567 Ki = 170 nM T57392 D0IA9Y 53472683 IC50 > 40000 nM T57392 D0IQ0Z 46885626 IC50 = 12000 nM T57392 D0IZ8X 90111638 IC50 > 100000 nM T57392 D0J1HB 23063810 IC50 > 100000 nM T57392 D0JT5I 24771824 IC50 = 14500 nM T57392 D0K1EG 11508736 IC50 > 100000 nM T57392 D0K4JQ 57339460 IC50 > 33000 nM T57392 D0K5HI 5311424 IC50 = 18000 nM T57392 D0K7FY 72703790 IC50 = 7000 nM T57392 D0L9KH 44623998 IC50 > 50000 nM T57392 D0L9QM 59568713 IC50 > 50000 nM T57392 D0M4TJ 44219292 IC50 > 50000 nM T57392 D0M9RQ 11697697 IC50 > 27000 nM T57392 D0MR0B 54766013 IC50 > 10000 nM T57392 D0N5KS 154104 IC50 < 10000 nM T57392 D0N6NM 71721648 IC50 > 5600 nM T57392 D0N6SO 15983988 IC50 < 10000 nM T57392 D0O2XQ 11256587 IC50 = 1600 nM T57392 D0P0KN 16739650 IC50 = 950 nM T57392 D0PN8H 46216796 IC50 > 5000 nM T57392 D0PW4N 6851740 IC50 > 25000 nM T57392 D0Q0AP 10409068 IC50 > 40000 nM T57392 D0Q7NB 10253143 IC50 > 100000 nM T57392 D0QR5G 2355 IC50 > 10000 nM T57392 D0R3VK 42642654 IC50 > 10000 nM T57392 D0RL4X 45270144 IC50 > 30000 nM T57392 D0S0EQ 9951066 IC50 = 46000 nM T57392 D0S1XX 134821691 IC50 > 40000 nM T57392 D0S2PD 42634627 IC50 > 30000 nM T57392 D0S5IR 86294073 IC50 > 30000 nM T57392 D0SG7B 49831257 IC50 > 70000 nM T57392 D0SP5V 49843471 IC50 > 50000 nM T57392 D0T0PN 9821217 Ki = 20 nM T57392 D0T3DO 9867758 IC50 = 25000 nM T57392 D0T4SG 11292191 IC50 > 10000 nM T57392 D0U4FF 10437018 IC50 > 40000 nM T57392 D0U7KH 86567195 IC50 > 5000 nM T57392 D0V9VG 51049968 IC50 >= 20000 nM T57392 D0VI4N 90409366 IC50 > 10000 nM T57392 D0W1US 1684 IC50 = 1258.93 nM T57392 D0W8XT 60663 IC50 = 63 nM T57392 D0W9VW 11526696 IC50 = 84000 nM T57392 D0X7EG 11462174 IC50 > 30000 nM T57392 D0XD4I 118502708 IC50 > 30000 nM T57392 D0Y1NC 148198 IC50 = 190 nM T57392 D0Y7NA 49871007 IC50 > 25000 nM T57392 D0YB2Y 42641863 Ki > 30000 nM T57392 D0ZE1O 9949641 IC50 > 50000 nM T57392 D0LF0O 135441202 IC50 > 40000 nM T57392 D00OWF 5280953 Ki = 50000 nM T57392 D03ZXG 118103874 IC50 > 30000 nM T57392 D08DMM 91799365 IC50 > 30000 nM T57392 D08SNH 71555922 IC50 = 47000 nM T57392 D0D3GL 137662068 IC50 > 40000 nM T57392 D0G2TX 46911228 IC50 > 5000 nM T57392 D0HG2S 86294663 IC50 > 30000 nM T57392 D0LI2I 118096900 IC50 > 30000 nM T57392 D0LU9X 74221950 IC50 > 50000 nM T57392 D0N6HP 91886057 IC50 = 26500 nM T57392 D0NJ9E 118096899 IC50 > 30000 nM T57392 D0QE8S 60197821 IC50 > 30000 nM T57392 D0QZ8K 70874141 IC50 = 9500 nM T57392 D0TR9T 45256914 IC50 > 5000 nM T57392 D0W1XE 91827457 IC50 > 30000 nM T57392 D0WR7B 122650373 IC50 > 30000 nM T57392 D0ZM8H 25265637 IC50 > 20000 nM T57392 D01NJT 65856 IC50 = 3162.28 nM T57392 D01TBN 188927 Ki = 420 nM T57392 D03EZB 9864291 IC50 = 9200 nM T57392 D03YPJ 5163 IC50 = 30000 nM T57392 D04RLX 148201 IC50 = 100000 nM T57392 D04WCI 16220188 IC50 > 29000 nM T57392 D04YHW 11406590 IC50 > 40000 nM T57392 D05MCS 44473151 IC50 > 40000 nM T57392 D06BPG 4528 IC50 > 20000 nM T57392 D06TGE 11226090 IC50 = 0.59 nM T57392 D06ZVC 10150497 IC50 = 196000 nM T57392 D07EBU 135565424 IC50 > 15000 nM T57392 D07GIB 11614352 IC50 = 23000 nM T57392 D07XPE 8249 IC50 = 27000 nM T57392 D08QHS 11296282 IC50 > 10000 nM T57392 D08QTP 6478034 IC50 > 50000 nM T57392 D09EVZ 507806 IC50 > 40000 nM T57392 D09NBM 10417440 IC50 = 37000 nM T57392 D09VTB 71768520 IC50 >= 10000 nM T57392 D0A1NU 16049769 IC50 > 30000 nM T57392 D0B4TT 17747460 IC50 = 40 nM T57392 D0B7SP 11292933 IC50 = 86000 nM T57392 D0G1RH 6918446 IC50 = 0.045 nM T57392 D0G6SZ 3001322 IC50 > 30000 nM T57392 D0H9GQ 9795276 IC50 = 780 nM T57392 D0IP6X 219077 IC50 = 55000 nM T57392 D0L5UO 9939609 IC50 = 26000 nM T57392 D0N8NK 11641563 IC50 > 10000 nM T57392 D0R7GH 9833312 IC50 = 4400 nM T57392 D0Y2HR 2247 IC50 > 30000 nM T57392 D0YE2N 73214 IC50 > 20000 nM T57392 CHV5M7 3634 IC50 = 1500 nM T57392 C9LCD8 3823 IC50 = 16300 nM T57392 C2KJI7 3883 IC50 = 2900 nM T57392 CS0ZC5 6768 Ki = 720 nM T57392 CNA29Q 7047 Ki > 1000000 nM T57392 C5RP9K 10651 Ki = 4000 nM T57392 CT34EY 12835 Ki = 100000 nM T57392 CKJ48S 14860 Ki > 1000000 nM T57392 C59DKW 15381 Ki > 1000000 nM T57392 CN0WP7 15630 IC50 < 10000 nM T57392 C7H2NQ 21138 IC50 = 1900 nM T57392 C6GN7M 40692 IC50 > 30000 nM T57392 C65PNO 41446 IC50 = 18100 nM T57392 CIX8D1 55750 IC50 = 8700 nM T57392 CK6VT0 60923 IC50 = 11 nM T57392 C2FVG0 64149 IC50 > 30000 nM T57392 CL15AQ 65373 IC50 > 100000 nM T57392 CMLI08 68079 IC50 > 10000 nM T57392 C1B9ZO 68094 Ki = 65000 nM T57392 C95JWC 68487 IC50 > 300000 nM T57392 C06GWQ 72340 Ki = 1100 nM T57392 C0VNL1 73391 Ki = 2200 nM T57392 CO0HB3 75473 Ki > 400000 nM T57392 C7SXL6 87152 IC50 > 25000 nM T57392 C96RZY 90454 IC50 = 1800 nM T57392 CB6G3Z 91536 IC50 = 1400 nM T57392 CA12VF 92390 IC50 = 1017000 nM T57392 CC0P7F 94378 IC50 > 30000 nM T57392 CYU2P9 98570 Ki = 122 nM T57392 CZB67X 98608 IC50 > 10000 nM T57392 C4WFM6 100146 IC50 = 1600 nM T57392 CP38TV 100267 IC50 = 11000 nM T57392 CXK76V 100580 IC50 = 196000 nM T57392 C0K7OY 108137 IC50 = 82000 nM T57392 CEP43C 122068 IC50 = 6400 nM T57392 C6QB9N 126266 IC50 = 4930 nM T57392 CY9T2A 127360 IC50 = 80 nM T57392 C6UXJ5 136621 IC50 > 1000000 nM T57392 CM2H7V 152430 IC50 > 10000 nM T57392 C5C2BD 156418 IC50 < 100 nM T57392 CL54TG 160521 IC50 = 97700 nM T57392 CK8RD5 168114 IC50 = 42700 nM T57392 CJ34CF 168115 IC50 = 54900 nM T57392 CDB9P5 170922 IC50 < 10000 nM T57392 C4RFP5 179460 Ki = 17 nM T57392 CA91IX 185559 Ki = 78 nM T57392 C1R6GB 189060 IC50 > 10000 nM T57392 CVL3Z7 190901 IC50 = 46 nM T57392 C0B5GC 224604 IC50 = 2200 nM T57392 CYS4H5 230263 IC50 = 8000 nM T57392 CIR36G 275548 IC50 = 570000 nM T57392 CJ6S0Z 285510 IC50 = 7300 nM T57392 C3ZT2Q 301389 IC50 = 2021000 nM T57392 CPK5E0 323023 IC50 = 83000 nM T57392 CLR67M 330747 IC50 = 8500 nM T57392 CAM18T 332425 IC50 > 100000 nM T57392 C9DG0W 332427 IC50 > 100000 nM T57392 CAS18T 359052 IC50 > 30000 nM T57392 CIXO41 408043 IC50 = 2100 nM T57392 CGA85T 408974 IC50 = 3500 nM T57392 CDU5O6 421105 IC50 = 1000 nM T57392 CCS9U7 424326 IC50 = 554000 nM T57392 CB08EU 425818 IC50 = 2400 nM T57392 CCX31R 428490 IC50 = 169000 nM T57392 CLD6J9 441074 IC50 = 2 nM T57392 C5Q8IX 457194 IC50 = 17700 nM T57392 C2K7AC 465996 IC50 = 1300 nM T57392 CVH49X 480768 IC50 > 20000 nM T57392 CRH1D7 491206 IC50 = 4000 nM T57392 C3Q0TX 493820 IC50 = 2430 nM T57392 CUO16L 493830 IC50 520 nM T57392 CKC8U4 507751 IC50 > 40000 nM T57392 CPXL01 507783 IC50 = 38000 nM T57392 CM40AT 507791 IC50 > 40000 nM T57392 C18QJF 515047 IC50 = 27000 nM T57392 CEN81S 515051 IC50 = 27000 nM T57392 CHX85A 515052 IC50 > 30000 nM T57392 CV6Y9X 550909 IC50 = 310 nM T57392 C2Y4TD 577307 IC50 > 40000 nM T57392 C6R5XN 595145 IC50 > 400000 nM T57392 CVRM18 595254 Ki = 124000 nM T57392 CR98MZ 613528 IC50 > 30000 nM T57392 C4FC1N 626798 IC50 > 50000 nM T57392 CX5V2H 636822 IC50 > 100000 nM T57392 CS5PK2 640180 IC50 = 68500 nM T57392 C03GIF 656862 IC50 = 20 nM T57392 CTGL43 672443 IC50 = 50000 nM T57392 CGL5R1 683949 IC50 = 8790 nM T57392 CN5CJ7 688803 IC50 > 10000 nM T57392 C2AHB4 689051 IC50 > 10000 nM T57392 C74MRA 702869 IC50 = 4280 nM T57392 C3LU7J 736282 Ki = 120 nM T57392 C6DJ3Y 741004 IC50 = 1230 nM T57392 CSUL21 780263 IC50 = 1360 nM T57392 CP23UY 780805 IC50 > 30000 nM T57392 CI43WJ 802727 IC50 > 10000 nM T57392 C3LM4S 821286 IC50 = 50 nM T57392 C06WCN 827839 IC50 = 90 nM T57392 C90NZF 853261 IC50 = 3000 nM T57392 CYKE37 863679 IC50 > 20000 nM T57392 CLJU94 877119 IC50 = 10000 nM T57392 C2TDG1 883547 IC50 > 40000 nM T57392 CB3V6I 929273 Ki = 6300 nM T57392 CMOR75 945544 IC50 = 6000 nM T57392 CMO9N5 970725 IC50 > 30000 nM T57392 CZG18E 1201554 Ki > 400000 nM T57392 CAZT67 1283333 IC50 = 100000 nM T57392 CV0Q3D 1302369 IC50 = 21200 nM T57392 C5G4FA 1394668 IC50 = 6000 nM T57392 C0GE2X 1619763 IC50 = 8130 nM T57392 C21HKV 1941609 IC50 > 30000 nM T57392 C3LSW0 2088634 IC50 > 50000 nM T57392 CZL8R3 2187415 IC50 > 50000 nM T57392 CP53EV 2350190 IC50 = 11000 nM T57392 CQTY36 2650025 IC50 = 1940 nM T57392 CZY89U 2727594 IC50 = 83900 nM T57392 CD28JA 2735964 IC50 > 25000 nM T57392 C5T3HX 2748785 IC50 > 10000 nM T57392 C0ZI1F 2756534 IC50 > 30000 nM T57392 CT6P3F 2782903 IC50 > 30000 nM T57392 CF2N8O 2794167 IC50 > 30000 nM T57392 C2LF9Q 2813098 Ki = 5500 nM T57392 CTBC06 2941086 IC50 = 10000 nM T57392 C14NBG 3008866 IC50 = 4800 nM T57392 C4XNG5 3012020 IC50 > 30000 nM T57392 C6TO5V 3012027 IC50 > 30000 nM T57392 CCQI26 3012527 IC50 = 50000 nM T57392 CM70GI 3013843 IC50 > 100000 nM T57392 CQ2SG0 3031421 IC50 > 20000 nM T57392 CAJQ53 3040177 IC50 = 98000 nM T57392 CT2WK9 3058605 Ki = 31 nM T57392 C82XOE 3083746 IC50 > 100000 nM T57392 C3F0GS 3120536 IC50 > 10000 nM T57392 C7CUZ5 3123921 IC50 = 28000 nM T57392 CFPR85 3213696 IC50 > 5000 nM T57392 C23VGA 3449946 IC50 = 30000 nM T57392 CI30FE 3463042 IC50 > 40000 nM T57392 CSW59H 3718258 IC50 > 100000 nM T57392 CK93HP 3844414 IC50 = 2900 nM T57392 CO23EI 3959338 IC50 > 20000 nM T57392 C1ZC4D 4384047 IC50 = 120 nM T57392 CE0OD3 4652320 IC50 > 40000 nM T57392 CZO2E5 4674678 IC50 = 13150 nM T57392 CFL8J3 4786512 IC50 = 100 nM T57392 CBFV62 4817293 IC50 = 11600 nM T57392 CJ8PL6 4840815 IC50 = 32000 nM T57392 CZU2N7 4862343 IC50 = 6000 nM T57392 C16EGI 4961254 IC50 > 10000 nM T57392 C80NAU 5273742 IC50 = 30000 nM T57392 C2BQN6 5281304 IC50 = 514000 nM T57392 CE6IV2 5281404 Ki = 86000 nM T57392 CZM7D8 5281794 IC50 = 87000 nM T57392 CA5D1J 5289110 IC50 > 20000 nM T57392 CZ09MD 5299617 IC50 = 9400 nM T57392 CMBL90 5300578 IC50 = 20000 nM T57392 CC49SG 5316673 IC50 > 100000 nM T57392 CA7UL5 5329333 IC50 > 50000 nM T57392 COQ41S 5329336 IC50 > 100000 nM T57392 COJI90 5338258 IC50 > 10000 nM T57392 CWFP51 5338324 IC50 = 12000 nM T57392 CU47YI 5351283 IC50 = 288000 nM T57392 CN0R5K 5352001 IC50 = 45500 nM T57392 C5Z0HQ 5355549 IC50 = 8200 nM T57392 C1D0RN 5470187 IC50 > 100000 nM T57392 CB4A3U 5481990 Ki = 32000 nM T57392 C3Q2XB 5495793 IC50 = 17000 nM T57392 C0ZAM9 5495818 IC50 = 9700 nM T57392 CPT10H 5717399 IC50 = 14000 nM T57392 C21EJH 5717404 IC50 = 1100 nM T57392 CE9KZ5 5720628 IC50 = 7700 nM T57392 CJMQ48 5737900 IC50 = 14000 nM T57392 CSH9C1 5787676 IC50 = 14000 nM T57392 CMWC08 5837372 IC50 > 10000 nM T57392 CAJK62 5859537 IC50 = 11000 nM T57392 CX23PO 6020016 IC50 > 10000 nM T57392 C2V8QP 6174007 IC50 = 1740 nM T57392 CTG9I2 6258621 IC50 = 1000 nM T57392 CR8P9W 6262995 IC50 > 10000 nM T57392 CA74LD 6320546 IC50 > 30000 nM T57392 C97UBE 6432105 Ki = 66 nM T57392 CGJ16S 6436013 IC50 > 5000 nM T57392 CB75NI 6479949 IC50 > 30000 nM T57392 C09BQE 6479956 IC50 = 30000 nM T57392 CEL6U1 6479971 IC50 = 30000 nM T57392 CC6U7A 6493950 IC50 < 1000 nM T57392 CN0VB3 6914627 IC50 > 30000 nM T57392 C80XWJ 6914629 IC50 > 30000 nM T57392 C0QCK1 6918455 IC50 = 32000 nM T57392 C48OIX 7074967 Ki = 165000 nM T57392 CU68IK 7141881 IC50 > 10000 nM T57392 CWX15G 7514880 IC50 = 10200 nM T57392 CJH57U 8854335 IC50 = 10000 nM T57392 C2W6PI 8867347 IC50 > 15000 nM T57392 C5J8HN 8902499 IC50 = 10200 nM T57392 C3EQL0 8931830 IC50 = 74200 nM T57392 C24MJV 9554928 IC50 = 23300 nM T57392 C32HVW 9554933 IC50 > 100000 nM T57392 CIA9B5 9794218 IC50 = 60700 nM T57392 C6YDQ0 9795278 IC50 > 3000 nM T57392 CA15IT 9796590 IC50 > 30000 nM T57392 CUGX54 9797385 IC50 = 15000 nM T57392 CVZG73 9799417 IC50 > 200000 nM T57392 CMIW83 9812710 IC50 > 30000 nM T57392 CR8ET5 9814387 IC50 = 2700 nM T57392 C1H7KW 9814761 IC50 > 30000 nM T57392 CFW74D 9815391 IC50 > 100000 nM T57392 CTN13P 9820134 IC50 = 300 nM T57392 C1E2DV 9826083 IC50 > 2000 nM T57392 C3NO4W 9828630 IC50 > 30 nM T57392 C2XA5B 9835305 IC50 > 30000 nM T57392 C13FZK 9849910 Ki = 550 nM T57392 CL79YZ 9858476 IC50 = 1700 nM T57392 CDQ91J 9862335 IC50 = 100 nM T57392 CSTG23 9866745 IC50 = 500 nM T57392 CN9YD5 9868131 IC50 = 45 nM T57392 CI6V2U 9870337 IC50 = 3900 nM T57392 CKF09P 9871544 IC50 = 6500 nM T57392 CQ4LC2 9872676 IC50 > 30000 nM T57392 CTZP28 9875352 IC50 = 360 nM T57392 COCP14 9879332 IC50 = 2000 nM T57392 CBF9T3 9879532 IC50 = 400 nM T57392 C7WCB6 9883332 IC50 > 30000 nM T57392 C1ZF0K 9886775 Ki = 600 nM T57392 CJW1P5 9888494 IC50 = 10000 nM T57392 CFRS47 9910748 IC50 = 1200 nM T57392 C4B2QY 9913339 IC50 > 20000 nM T57392 C5T7UK 9921294 IC50 = 400 nM T57392 C9MDU2 9921865 IC50 = 5000 nM T57392 C29WVT 9923385 IC50 > 25000 nM T57392 CX5GL1 9928224 IC50 = 40 nM T57392 C0C7NV 9930121 IC50 > 10000 nM T57392 C10VOI 9930235 IC50 = 76 nM T57392 CGL13H 9939495 IC50 = 24000 nM T57392 CFC48H 9940105 IC50 = 15600 nM T57392 COD73F 9943346 IC50 = 3600 nM T57392 C02XPN 9944222 IC50 > 30000 nM T57392 CEB1I2 9945500 IC50 > 25000 nM T57392 CIHX05 9946012 IC50 > 30000 nM T57392 CG9KR4 9948238 IC50 = 30 nM T57392 CMI58L 9956563 IC50 = 3 nM T57392 CNJ81W 9959174 IC50 = 14000 nM T57392 CY9Q2M 9966187 IC50 = 4100 nM T57392 C7ZK5J 9966516 IC50 > 14000 nM T57392 CKLH03 9967123 IC50 = 1700 nM T57392 CBV8L2 9968207 IC50 > 30000 nM T57392 CMY73F 9978490 IC50 = 6000 nM T57392 CGEJ24 9985625 IC50 > 100000 nM T57392 C9Y6GX 9985634 IC50 = 2000 nM T57392 C98KZE 10002960 IC50 = 1700 nM T57392 C26QHZ 10005638 IC50 > 2000 nM T57392 CCD24K 10007859 IC50 >= 18000 nM T57392 C0KHW3 10022393 IC50 > 100000 nM T57392 C5TRX2 10025406 IC50 = 1500 nM T57392 CA06TQ 10028888 IC50 > 100000 nM T57392 C47DPZ 10030750 IC50 > 30000 nM T57392 C1WH8Q 10042344 IC50 > 40000 nM T57392 CGNA89 10045603 IC50 = 22000 nM T57392 CPI2Q0 10049358 IC50 = 27000 nM T57392 CK63CE 10050884 Ki = 2600 nM T57392 CSOR04 10070428 IC50 = 51000 nM T57392 C5B4HJ 10071498 IC50 > 100000 nM T57392 CL8WC4 10075685 IC50 > 30000 nM T57392 CVE2T1 10076176 IC50 = 6400 nM T57392 CJO8N5 10088963 IC50 = 68100 nM T57392 C1XH8C 10091613 IC50 = 8800 nM T57392 C2G3MJ 10099429 IC50 > 30000 nM T57392 CEA01V 10108128 IC50 = 410 nM T57392 C1TY3F 10122289 IC50 = 6000 nM T57392 C0KOC5 10122452 IC50 = 83000 nM T57392 C1LSI8 10122657 IC50 = 9000 nM T57392 CC2YT5 10122981 IC50 = 29600 nM T57392 C6HR7P 10130125 IC50 > 100000 nM T57392 C47RHT 10130685 IC50 = 32000 nM T57392 CIU8H6 10131483 IC50 > 30000 nM T57392 CD75GU 10131619 IC50 > 10000 nM T57392 CRW07C 10133485 IC50 = 35800 nM T57392 CP64RT 10134089 IC50 > 10000 nM T57392 CPH1C7 10140602 IC50 = 4400 nM T57392 CR6H9Y 10146899 IC50 = 530 nM T57392 COFT51 10154555 IC50 = 3200 nM T57392 CQO8H3 10157813 IC50 > 30000 nM T57392 C1VQ4M 10162564 IC50 = 1300 nM T57392 CLT63F 10166543 IC50 > 50000 nM T57392 CJ4R2U 10168216 IC50 = 25000 nM T57392 CP6Q1W 10173403 IC50 = 1500 nM T57392 CAK3E1 10189993 IC50 = 22000 nM T57392 CDP14A 10190433 IC50 = 12000 nM T57392 CEDW91 10190506 IC50 = 8800 nM T57392 CA4N2V 10198034 IC50 > 100000 nM T57392 CM0F5B 10198293 IC50 = 93500 nM T57392 CG6IF7 10212348 IC50 = 14900 nM T57392 C8DWX5 10219789 IC50 > 100000 nM T57392 CX32UD 10223809 IC50 = 42000 nM T57392 CV5X8A 10224181 IC50 > 2500 nM T57392 C4JN9U 10224745 IC50 > 50000 nM T57392 CFQ5L2 10232552 IC50 = 15000 nM T57392 CB72SI 10233112 IC50 = 39000 nM T57392 C9UIX5 10233517 IC50 = 39000 nM T57392 C1B7ZE 10233723 IC50 = 19000 nM T57392 CKE5C6 10233724 IC50 = 3600 nM T57392 CN4G5C 10244716 IC50 = 600 nM T57392 CFZQ39 10249083 IC50 = 13000 nM T57392 CK73CO 10267677 IC50 > 30000 nM T57392 C4KU1Y 10268204 IC50 > 25000 nM T57392 CU1ZW4 10268255 IC50 = 1300 nM T57392 C2EO1A 10273854 IC50 = 33000 nM T57392 CE9ID0 10280944 IC50 = 7800 nM T57392 C61ZEV 10282620 IC50 = 14000 nM T57392 CWOR29 10283706 IC50 = 6400 nM T57392 CO38FQ 10283896 IC50 = 22200 nM T57392 C16MNJ 10284289 IC50 < 1000 nM T57392 CO2LT5 10286610 IC50 > 40000 nM T57392 C7C5FN 10294289 IC50 = 4400 nM T57392 CE4Y7G 10294290 IC50 > 30000 nM T57392 C3FL9K 10295633 IC50 > 2000 nM T57392 CO0P4F 10301330 IC50 = 4600 nM T57392 CQV98P 10305047 IC50 = 24000 nM T57392 C7W2NF 10305573 IC50 = 56000 nM T57392 C9C3KH 10305705 IC50 = 11100 nM T57392 CAU47H 10305883 IC50 = 10500 nM T57392 CD3ER5 10308589 IC50 > 50000 nM T57392 C6ITS2 10313487 IC50 > 100000 nM T57392 CZ18PL 10316203 IC50 = 3000 nM T57392 C8F1LK 10318708 IC50 > 100000 nM T57392 C27TCH 10319351 IC50 = 13000 nM T57392 CM46XO 10327211 IC50 = 3700 nM T57392 C4AJ0X 10341839 IC50 = 45000 nM T57392 C63GNX 10342726 IC50 = 5526 nM T57392 CFXA48 10343679 IC50 > 25000 nM T57392 CW50TU 10345610 IC50 > 30000 nM T57392 CQVP17 10347783 IC50 > 50000 nM T57392 CPD85J 10347896 IC50 > 30000 nM T57392 CH38EM 10353296 IC50 = 86350 nM T57392 CW9P2U 10364379 IC50 > 100000 nM T57392 C4A5SP 10379988 IC50 = 5000 nM T57392 CA8B5T 10390073 IC50 > 2000 nM T57392 C5VAB7 10401590 IC50 = 1200 nM T57392 C3A2NK 10402335 Ki = 8000 nM T57392 CWK4O1 10406239 IC50 >= 5000 nM T57392 C8K7VS 10410589 IC50 > 100000 nM T57392 C6RVC0 10426237 IC50 = 600 nM T57392 CZ6SJ2 10435152 Ki = 7000 nM T57392 C18MRG 10436237 IC50 > 30000 nM T57392 CLDM93 10445840 IC50 > 10000 nM T57392 C97LHV 10454092 IC50 < 100 nM T57392 C9ODF7 10454589 IC50 > 100000 nM T57392 C8DWH6 10456892 IC50 > 30000 nM T57392 CJ1D7B 10458839 Ki = 2000 nM T57392 C1H5RP 10458842 IC50 > 10000 nM T57392 CFIE04 10459196 IC50 = 50500 nM T57392 C0FE3Q 10475883 IC50 = 14000 nM T57392 C8TPU0 10510985 Ki > 400000 nM T57392 C4CRA8 10624340 IC50 > 100000 nM T57392 C6UX4J 10633725 IC50 = 15000 nM T57392 CJPW17 10654534 Ki > 400000 nM T57392 CA82YQ 10704488 IC50 = 16000 nM T57392 C9SWF5 10791993 IC50 = 118576874.8 nM T57392 CXK63D 10829689 IC50 = 13200 nM T57392 CBK06L 10861643 IC50 = 291000 nM T57392 CZS9Q5 10899427 IC50 > 400000 nM T57392 C8U9GH 10927016 Ki = 1420 nM T57392 CH61UW 11128957 IC50 = 11000 nM T57392 CW1Q6S 11148656 IC50 = 1010 nM T57392 CCD91J 11148936 IC50 = 39800 nM T57392 CXT8Y2 11151568 IC50 < 10000 nM T57392 CB47FY 11154357 IC50 = 55000 nM T57392 C5K4PC 11160258 IC50 > 100000 nM T57392 C9AT4X 11163693 IC50 > 20000 nM T57392 C1A8HL 11171679 Ki = 127000 nM T57392 CP1EI3 11172276 IC50 = 7810 nM T57392 CJEW09 11176034 IC50 = 44200 nM T57392 CRU5Y3 11183547 IC50 > 100000 nM T57392 CY57GR 11187635 IC50 > 50000 nM T57392 CYB1W9 11187925 IC50 = 21100 nM T57392 CF86JN 11188632 IC50 = 300 nM T57392 C0XCD3 11195292 IC50 = 940 nM T57392 C7F6CE 11195591 IC50 = 96500 nM T57392 CHM83A 11199490 IC50 = 4100 nM T57392 CE6HS7 11200189 IC50 = 43000 nM T57392 C7U4SP 11203112 IC50 > 100000 nM T57392 C1XR3I 11206290 Ki = 84500 nM T57392 CJ1O6V 11207072 IC50 = 36300 nM T57392 CV1SD9 11208566 IC50 > 10000 nM T57392 CIAE47 11211122 IC50 = 30000 nM T57392 C4O3QM 11218177 IC50 = 53300 nM T57392 CIB34F 11218910 IC50 > 100000 nM T57392 CI2SN0 11222420 IC50 > 25000 nM T57392 CA39QR 11227406 IC50 = 30 nM T57392 CEW9L6 11228293 IC50 > 5000 nM T57392 CMHY80 11229234 Ki = 45300 nM T57392 CA71OC 11235004 IC50 > 100000 nM T57392 C9WY6K 11235389 IC50 > 50000 nM T57392 C6D3UR 11237434 IC50 > 30000 nM T57392 C8IQ7N 11247557 IC50 = 24000 nM T57392 CMFI07 11248182 IC50 = 1500 nM T57392 CLR09Q 11253245 IC50 > 100000 nM T57392 CWZP56 11256722 IC50 = 4100 nM T57392 C5NCH0 11258701 IC50 = 190 nM T57392 C7KU1G 11264664 IC50 = 500 nM T57392 C92CYH 11265950 IC50 = 6679 nM T57392 CRZ3V0 11269310 IC50 = 2600 nM T57392 CQ6KW0 11272103 IC50 = 200 nM T57392 C9W2NY 11274374 IC50 > 10000 nM T57392 C9W4KE 11275964 IC50 = 6000 nM T57392 CA93LY 11280087 IC50 = 530 nM T57392 CG82EM 11280808 IC50 = 670 nM T57392 COV2U9 11281200 IC50 = 160 nM T57392 CQ2AW4 11299991 IC50 > 100000 nM T57392 CV1LG4 11301893 IC50 = 30000 nM T57392 C5CK3W 11304200 IC50 = 3400 nM T57392 CBEW43 11308052 IC50 > 50000 nM T57392 CF5YS9 11310529 Ki = 14400 nM T57392 CK8L6D 11310871 IC50 > 100000 nM T57392 CB7YS1 11315814 IC50 > 5000 nM T57392 C8S4FU 11317045 IC50 > 29100 nM T57392 CO8B7R 11317439 IC50 > 25000 nM T57392 CMQD35 11321674 Ki = 56500 nM T57392 C7WA0E 11322127 IC50 = 398 nM T57392 CY9KM7 11322128 IC50 = 88700 nM T57392 CT6CH4 11322177 IC50 = 21400 nM T57392 CW01KR 11322201 IC50 > 100000 nM T57392 C1A5ET 11329244 IC50 = 240 nM T57392 C7O0ER 11337925 IC50 = 6200 nM T57392 CU72EY 11344157 Ki = 102000 nM T57392 CPK71M 11345209 IC50 = 6590 nM T57392 CPSQ49 11350705 IC50 = 760 nM T57392 C5FG8X 11355925 IC50 > 400000 nM T57392 C84IUF 11357143 IC50 > 100000 nM T57392 C7I4FX 11363702 IC50 > 10000 nM T57392 C7DUQ5 11364979 IC50 = 43300 nM T57392 C8N0GX 11368215 IC50 = 120 nM T57392 CI5GZ4 11368318 IC50 > 100000 nM T57392 CGT16B 11372452 IC50 = 5300 nM T57392 CC0L7O 11377200 IC50 > 50000 nM T57392 C1BOK3 11378800 Ki = 96500 nM T57392 C0YO8L 11378954 IC50 = 85500 nM T57392 CD82VI 11379226 IC50 = 81600 nM T57392 CD68AR 11380674 IC50 < 50 nM T57392 C2E8MJ 11382472 IC50 = 89 nM T57392 CX5Z0G 11383671 IC50 = 700 nM T57392 CZIC23 11389737 IC50 = 199000 nM T57392 CYL06Q 11389927 IC50 = 296000 nM T57392 CKZV96 11393842 IC50 > 100000 nM T57392 C9AOM3 11397017 IC50 > 10000 nM T57392 CQE92F 11406708 IC50 = 9500 nM T57392 C1COT8 11408302 IC50 = 9600 nM T57392 CN6G8I 11408550 IC50 = 8700 nM T57392 C0N5JW 11408724 IC50 = 4200 nM T57392 CMW42X 11416123 IC50 > 20000 nM T57392 CLR3W7 11424804 IC50 = 10800 nM T57392 CML2H3 11428837 IC50 = 4300 nM T57392 CVBO48 11428892 IC50 = 3000 nM T57392 C3PSN6 11429436 IC50 = 3400 nM T57392 CUSQ84 11430331 IC50 = 16000 nM T57392 CKL6P9 11440457 IC50 > 10000 nM T57392 CMH9J5 11450298 IC50 = 4800 nM T57392 C3CU1H 11450354 IC50 > 40000 nM T57392 CX3ZU0 11450539 IC50 = 100 nM T57392 CE42DM 11453673 IC50 = 97800 nM T57392 CR4IV6 11453965 IC50 = 8000 nM T57392 CPIH90 11458616 IC50 = 9540 nM T57392 CX4K6J 11463076 IC50 = 2500 nM T57392 C7IXL1 11463580 IC50 = 8600 nM T57392 C24ZHJ 11463610 IC50 > 10000 nM T57392 CR4N5I 11465834 IC50 = 66000 nM T57392 CAO2E4 11465947 IC50 = 5400 nM T57392 C5GOD3 11477039 IC50 = 9000 nM T57392 CW57BU 11480732 IC50 = 344000 nM T57392 C69PFD 11484605 IC50 = 32000 nM T57392 C4R8HV 11485758 IC50 = 510 nM T57392 COC7Q9 11488952 IC50 = 62000 nM T57392 C1O9XD 11493620 IC50 > 10000 nM T57392 CW3YO5 11494768 IC50 > 50000 nM T57392 C69AMJ 11500781 IC50 = 5500 nM T57392 C3B0LO 11501191 IC50 = 65 nM T57392 CTYJ07 11501580 IC50 = 21000 nM T57392 CYC7D5 11503034 IC50 = 7200 nM T57392 CFSH67 11504490 IC50 > 10000 nM T57392 CLPO39 11508317 IC50 = 2700 nM T57392 CQ6IU7 11509269 IC50 > 10000 nM T57392 CDQ18N 11515125 IC50 = 2 nM T57392 CP9RB7 11515387 IC50 = 320 nM T57392 C0SN2O 11515728 IC50 > 10000 nM T57392 COTH53 11516139 IC50 = 5300 nM T57392 CX4MA8 11519486 IC50 > 40000 nM T57392 CY47AQ 11519784 IC50 > 10000 nM T57392 CVO7T9 11522969 IC50 > 10000 nM T57392 C7HNP0 11526745 IC50 = 31000 nM T57392 C0BF5R 11527661 IC50 > 25000 nM T57392 C75FPD 11529874 IC50 = 1860 nM T57392 CR92GA 11537005 IC50 = 970 nM T57392 CF2OM8 11539410 IC50 > 50000 nM T57392 C0ZF8J 11544156 IC50 = 200 nM T57392 C3VP9T 11544537 IC50 > 10000 nM T57392 C7IOJ0 11548023 IC50 = 5200 nM T57392 C34JAV 11551351 IC50 = 3300 nM T57392 C3RMI1 11559300 IC50 > 30000 nM T57392 CY5NE2 11559695 IC50 = 100 nM T57392 C0H8CM 11561655 IC50 = 4500 nM T57392 C84NIF 11566130 IC50 > 10000 nM T57392 C1VF0P 11566266 IC50 = 290 nM T57392 CDFU34 11566489 IC50 > 10000 nM T57392 CB59HM 11570626 IC50 > 100000 nM T57392 C4IX6W 11573549 IC50 > 10000 nM T57392 CMX60P 11573849 IC50 = 17600 nM T57392 CR75FZ 11577204 IC50 > 30000 nM T57392 CXP2M0 11580426 IC50 = 6900 nM T57392 CW7G3X 11580427 IC50 = 28000 nM T57392 CVX6K7 11580514 IC50 > 10000 nM T57392 C3YXZ7 11582291 IC50 = 30000 nM T57392 CFZ1Q5 11584681 IC50 > 40000 nM T57392 CFU15B 11588489 IC50 = 89000 nM T57392 C1HG4A 11591164 IC50 = 91000 nM T57392 CV9B8R 11595360 IC50 < 50 nM T57392 CHU90R 11598626 IC50 > 8000 nM T57392 CP56DO 11599295 IC50 > 10000 nM T57392 C15TEH 11604449 IC50 > 10000 nM T57392 CPH40V 11607042 IC50 > 30000 nM T57392 CH7P9Z 11608743 IC50 > 30000 nM T57392 C7ENB2 11609939 IC50 = 21500 nM T57392 C6HLN8 11610150 IC50 = 5540 nM T57392 C2M8HZ 11610353 IC50 > 50000 nM T57392 CKXH63 11610910 IC50 > 12000 nM T57392 C5JZ6R 11615459 IC50 > 40000 nM T57392 CW0ZM6 11619260 IC50 = 5000 nM T57392 C5FQR2 11622909 IC50 = 31622.78 nM T57392 C79OMR 11623756 IC50 = 7300 nM T57392 C1KD4Z 11623823 IC50 = 21800 nM T57392 CSB9O5 11623845 IC50 = 856000 nM T57392 CGX96V 11626927 IC50 < 50118.72 nM T57392 C9L5VD 11631813 IC50 > 50000 nM T57392 C23XSL 11638166 Ki = 850 nM T57392 CCP69D 11638499 IC50 > 10000 nM T57392 CRT09O 11638500 IC50 > 10000 nM T57392 CQ1U9W 11638962 IC50 = 480 nM T57392 CJS28X 11641672 IC50 = 200 nM T57392 CQRB62 11641686 IC50 = 1200 nM T57392 C6Y4HR 11647548 IC50 > 30000 nM T57392 CMB6F9 11653874 IC50 > 50000 nM T57392 CB7P8J 11655677 IC50 > 100000 nM T57392 CX7FR8 11655728 IC50 > 9000 nM T57392 CM2T8F 11656187 IC50 = 5700 nM T57392 CH3N1I 11659592 IC50 = 5200 nM T57392 CF92SM 11659664 IC50 = 27100 nM T57392 C3E0TV 11663187 IC50 = 3700 nM T57392 C51UDK 11667741 IC50 > 10000 nM T57392 CXJ17M 11669364 IC50 > 100000 nM T57392 CIUJ01 11670392 IC50 > 50000 nM T57392 C0V7SU 11675388 IC50 > 10000 nM T57392 C72BNQ 11682521 IC50 > 50000 nM T57392 CY36RI 11688223 IC50 = 12000 nM T57392 CW4U3H 11688520 IC50 > 10000 nM T57392 C3WBU8 11689242 IC50 = 14000 nM T57392 C7Z0SX 11695591 IC50 = 7500 nM T57392 C9CM2R 11695689 IC50 > 50000 nM T57392 CP3G0Q 11695811 IC50 = 9600 nM T57392 COH3C4 11697546 IC50 = 90 nM T57392 C65TAC 11698513 IC50 = 6100 nM T57392 C5ECV1 11699447 IC50 > 35000 nM T57392 CBDC74 11702114 IC50 = 15000 nM T57392 CQ5P2F 11702115 IC50 = 12000 nM T57392 CO3U4B 11705008 IC50 > 20000 nM T57392 C78GTN 11709314 IC50 = 1500 nM T57392 CL4DS1 11709762 IC50 > 10000 nM T57392 C4M9AU 11710505 IC50 = 3370 nM T57392 CHK5I2 11712756 IC50 > 9000 nM T57392 CN5UX7 11713409 IC50 > 40000 nM T57392 CN2L4J 11716660 IC50 = 800 nM T57392 CL5S9K 11719046 IC50 > 5000 nM T57392 C07CUH 11719337 IC50 > 10000 nM T57392 CZY05V 11719421 IC50 = 25000 nM T57392 CX9VH0 11720815 IC50 > 10000 nM T57392 CYQ4O9 11723225 IC50 = 27000 nM T57392 C0Z5JS 11740023 IC50 = 48000 nM T57392 CG6SM0 11749794 IC50 = 3200 nM T57392 CG0YB2 11751828 IC50 > 10000 nM T57392 CC92YE 11755033 IC50 > 100000 nM T57392 C8D7BS 11771234 IC50 = 12605 nM T57392 CB36OJ 11771503 IC50 > 40000 nM T57392 C6TS4D 11773824 IC50 > 5000 nM T57392 C6A1LM 11786814 IC50 > 500000 nM T57392 CN8CP5 11817019 IC50 = 12550 nM T57392 CS7W2V 11848793 IC50 > 30000 nM T57392 CI6JQ5 11855008 IC50 = 151000 nM T57392 CL1FX0 11947758 IC50 > 30000 nM T57392 CT0H7I 11949628 IC50 = 9900 nM T57392 CK13QD 11953409 IC50 = 1300 nM T57392 CK2EZ6 11962967 IC50 > 100000 nM T57392 CH26TZ 11963255 IC50 > 100000 nM T57392 C5QB3M 11963972 IC50 = 2300 nM T57392 C8P9GD 11966041 IC50 > 10000 nM T57392 CYEN98 11977494 IC50 > 100000 nM T57392 CN5W3V 11978858 IC50 > 100000 nM T57392 CW8T4V 11978859 IC50 > 100000 nM T57392 C1T8XZ 11993865 Ki > 400000 nM T57392 CBZ83S 11993868 Ki > 400000 nM T57392 C7A1EZ 11993870 Ki = 29800 nM T57392 C4XP2N 11993872 Ki = 45400 nM T57392 CWT0S3 11993875 Ki > 400000 nM T57392 CR4YS2 11996303 IC50 = 8000 nM T57392 C7D1AY 11996304 IC50 = 3000 nM T57392 C1A2IB 12001199 IC50 > 100000 nM T57392 CJM8C3 12032282 Ki = 1000 nM T57392 C9RX1L 12108566 IC50 = 8700 nM T57392 C3XK1M 12445790 IC50 = 8400 nM T57392 C96LHY 12619618 IC50 = 30 nM T57392 CO3VP9 12619657 IC50 = 50 nM T57392 CO3HN1 13163256 IC50 = 52000 nM T57392 C7I9PF 13557523 Ki > 400000 nM T57392 C0FY4P 13615899 IC50 = 5000 nM T57392 C1G0EZ 13957609 IC50 = 2170 nM T57392 COF3L5 14054408 IC50 = 21000 nM T57392 CIF90V 14434140 IC50 = 4400 nM T57392 CXS7Y5 14825858 IC50 > 100000 nM T57392 CR54KX 14861225 IC50 > 100000 nM T57392 C9VYL5 15172937 IC50 > 100000 nM T57392 C3YRU7 15295578 IC50 = 3300 nM T57392 C4FY2P 15549736 Ki = 2100 nM T57392 C21ITW 15549737 Ki = 4250 nM T57392 CO19UA 15595033 Ki = 6664 nM T57392 C7X3CQ 15604497 IC50 > 25118.86 nM T57392 CT4RL1 15778480 IC50 = 387000 nM T57392 CBE59I 15940927 IC50 > 100000 nM T57392 C08NEU 15945881 IC50 > 10000 nM T57392 C79VQK 15950271 IC50 > 10000 nM T57392 C3BI9R 15951010 IC50 > 10000 nM T57392 CWH1A8 15951076 IC50 > 10000 nM T57392 C2ZYA6 15951338 IC50 = 3480 nM T57392 C1Q8IV 15951410 IC50 = 927 nM T57392 CW8M6S 15952123 IC50 = 2500 nM T57392 CL1E6O 15953860 IC50 = 13000 nM T57392 CUI7P4 15955613 IC50 < 1000 nM T57392 C3W8ZL 15981007 IC50 > 50000 nM T57392 CW6S0H 15981486 IC50 = 6200 nM T57392 C2D1KP 15983982 IC50 = 3170 nM T57392 C5ACW8 15984094 Ki = 450 nM T57392 CQJ7Y2 15985912 IC50 > 50118.72 nM T57392 CPR25X 15986917 IC50 > 100000 nM T57392 C5KW3L 15987108 IC50 = 41000 nM T57392 CCL59Z 16007088 IC50 = 1600 nM T57392 C08CSK 16007091 IC50 > 18000 nM T57392 CG5A7W 16013152 IC50 = 1200 nM T57392 CBMF65 16013184 IC50 > 50000 nM T57392 C6V4TG 16013186 IC50 > 50000 nM T57392 C20CRP 16040587 IC50 = 15000 nM T57392 C8ZP3G 16041292 IC50 = 29000 nM T57392 CDU1L0 16041411 IC50 > 60000 nM T57392 CI6L0N 16042459 IC50 = 300 nM T57392 CMZU26 16043268 IC50 = 6300 nM T57392 C29KFG 16045493 IC50 = 47400 nM T57392 CR78OW 16046124 IC50 = 10000 nM T57392 CU27FI 16049886 IC50 = 17000 nM T57392 CZC7L2 16049887 IC50 > 25000 nM T57392 CQ9U1Y 16051921 IC50 = 6100 nM T57392 C30UFT 16066811 IC50 > 50000 nM T57392 CFK8J5 16068056 IC50 > 10000 nM T57392 CQRU95 16070337 IC50 > 25000 nM T57392 C8E6CH 16070448 IC50 = 5000 nM T57392 CTIQ90 16071896 IC50 > 25000 nM T57392 CX2GC6 16071897 IC50 > 25000 nM T57392 CL4ON2 16072021 IC50 = 5000 nM T57392 CJU50N 16072099 IC50 > 100000 nM T57392 C8D0KF 16099905 IC50 = 17000 nM T57392 C2FXW0 16099923 IC50 = 151000 nM T57392 CC24LB 16110489 IC50 > 10000 nM T57392 CHR8G4 16122633 IC50 > 10000 nM T57392 C0S1VK 16122818 IC50 > 40000 nM T57392 CFYL31 16122898 IC50 > 50000 nM T57392 C9G8TZ 16124598 IC50 = 100000 nM T57392 C0J6CH 16125372 IC50 = 4700 nM T57392 CMN0P3 16125681 IC50 = 5300 nM T57392 C4BYI2 16125682 IC50 = 12000 nM T57392 C8FLH6 16202152 IC50 = 10000 nM T57392 CWJZ50 16223655 IC50 = 4 nM T57392 CDG38L 16223656 IC50 > 10 nM T57392 C3O7HD 16223851 IC50 = 2.6 nM T57392 C0D9KR 16223854 IC50 > 30 nM T57392 C5L1QM 16224456 IC50 > 30 nM T57392 CTH6W4 16292141 IC50 > 25000 nM T57392 CQ3HO2 16309462 IC50 = 3400 nM T57392 CVJ4O1 16654686 IC50 = 277000 nM T57392 C4QU0M 16654984 IC50 > 6000 nM T57392 CY6D1F 16656782 IC50 > 25000 nM T57392 C6P4BX 16656803 IC50 = 13800 nM T57392 C7X0TS 16659334 IC50 > 30000 nM T57392 CIBY49 16661548 IC50 = 22000 nM T57392 C45KPZ 16661549 IC50 = 31000 nM T57392 CH60SU 16661701 IC50 = 18000 nM T57392 CU9LS2 16661702 IC50 = 1600 nM T57392 CXL4Q3 16663122 IC50 > 100000 nM T57392 CK4FJ8 16664733 IC50 > 20000 nM T57392 C1UY8J 16666386 IC50 > 20000 nM T57392 CH0Q9T 16678616 IC50 = 35000 nM T57392 C4FUO7 16678620 IC50 > 50000 nM T57392 CDY08B 16678725 IC50 = 900 nM T57392 C1N8IL 16679518 IC50 = 4000 nM T57392 C0CF9G 16679612 IC50 = 22000 nM T57392 C8X6SN 16679614 IC50 > 50000 nM T57392 CH8A2G 16679616 IC50 > 50000 nM T57392 CBE9O8 16679617 IC50 > 50000 nM T57392 CQF5Y7 16679701 IC50 > 50000 nM T57392 CSK8N5 16679707 IC50 = 15000 nM T57392 CAPU50 16719554 IC50 = 13000 nM T57392 CN95DG 16719649 IC50 > 100000 nM T57392 C92NRU 16727109 IC50 > 150000 nM T57392 CG04RZ 16727123 IC50 = 4300 nM T57392 CAX2B7 16728787 IC50 = 9800 nM T57392 C0H8UN 16730109 IC50 > 40000 nM T57392 C9BC0L 16732000 IC50 > 40000 nM T57392 CBR95H 16739953 IC50 = 15000 nM T57392 CLY57P 16744597 IC50 > 40000 nM T57392 CA68OS 16744599 IC50 = 40000 nM T57392 CUI0X4 16744748 IC50 > 40000 nM T57392 CM3OV0 16745085 IC50 = 40000 nM T57392 C94MKR 16745086 IC50 = 29000 nM T57392 C5GY6N 16745241 IC50 = 40000 nM T57392 CW85LQ 16745311 IC50 = 17300 nM T57392 CC4L1M 16747701 IC50 > 22000 nM T57392 CK3WA5 16747712 IC50 = 1400 nM T57392 CW2SY5 16750291 IC50 > 10000 nM T57392 CIX7U2 16750304 IC50 > 10000 nM T57392 C5DKZ8 16956771 IC50 > 11000 nM T57392 CU42ZC 17244953 IC50 < 10000 nM T57392 C8D4PX 17408359 IC50 = 8000 nM T57392 C9C5TV 17751819 IC50 = 660 nM T57392 C8TKD5 17754437 IC50 > 100000 nM T57392 CAJ0S2 17754557 EC50 > 50000 nM T57392 CT5L0Q 17955460 IC50 < 1000 nM T57392 C87WIK 18104758 IC50 > 50000 nM T57392 CF9TW8 18414685 IC50 = 35000 nM T57392 CG93TR 18440026 IC50 > 50000 nM T57392 C9JD5Y 19360456 IC50 = 36 nM T57392 C2HFY3 19553304 IC50 = 8800 nM T57392 CKH72O 20115797 IC50 = 50000 nM T57392 CT2KW6 20548414 IC50 = 50 nM T57392 CR1K3H 20763282 IC50 = 32000 nM T57392 C8X0RI 20763372 IC50 > 100000 nM T57392 C8OHP4 20763385 IC50 > 100000 nM T57392 C6POY9 20763386 IC50 = 83000 nM T57392 CZBJ32 20763421 IC50 = 98000 nM T57392 C7OMR1 20763606 IC50 > 100000 nM T57392 C81JWV 20906619 IC50 = 3000 nM T57392 CHC4Q3 21064283 IC50 > 30000 nM T57392 C1CA6D 21070989 IC50 > 10000 nM T57392 CBX5O7 21074158 IC50 = 10000 nM T57392 CY9B5M 21257907 IC50 > 4000 nM T57392 C18TEI 21303363 IC50 > 30000 nM T57392 CK7HS6 21362416 IC50 = 36000 nM T57392 C8OHV9 21362425 IC50 > 100000 nM T57392 CO17PU 21635104 IC50 = 130 nM T57392 CO6E2Z 21717336 IC50 = 2300 nM T57392 C7KIJ3 21717337 IC50 = 1100 nM T57392 CM1IF8 21914519 IC50 > 100000 nM T57392 CZF82E 21914667 IC50 > 63095.73 nM T57392 CK8X7S 21956341 IC50 = 4800 nM T57392 CZK6M0 22239024 IC50 = 90 nM T57392 CO32YX 22254068 IC50 > 10000 nM T57392 C4YP8N 22431956 IC50 = 20000 nM T57392 C9N5XW 22520172 IC50 = 5700 nM T57392 CIC7F6 22675312 IC50 = 1500 nM T57392 CP41JS 22675387 IC50 < 400 nM T57392 C5R7JT 22675398 IC50 = 1400 nM T57392 C0F3DZ 23330544 IC50 = 30 nM T57392 C3TVL7 23501721 IC50 > 7500 nM T57392 C8ZD9W 23567095 IC50 = 4200 nM T57392 C9NI1F 23567109 IC50 = 250 nM T57392 CZQP15 23567112 IC50 = 5400 nM T57392 C10UWF 23567114 IC50 = 5700 nM T57392 CIPX37 23567116 IC50 = 3900 nM T57392 CCT6R7 23567120 IC50 = 1100 nM T57392 CNH40T 23567127 IC50 = 760 nM T57392 C1Y8CH 23567131 IC50 = 5000 nM T57392 CJD8Q6 23567134 IC50 > 10000 nM T57392 C54SJG 23567138 IC50 = 1200 nM T57392 CF81SW 23582412 IC50 > 100000 nM T57392 C9K1DY 23583191 IC50 > 100000 nM T57392 C3K6HV 23594220 IC50 = 5792 nM T57392 CVBM54 23594222 IC50 = 1108 nM T57392 CXC6E3 23594223 IC50 = 4337 nM T57392 CQ93SH 23594225 IC50 = 7888 nM T57392 C4JGI8 23594247 IC50 = 5653 nM T57392 CW2R4M 23624283 IC50 = 54000 nM T57392 CO1NA8 23624297 IC50 = 26400 nM T57392 CQ29HW 23626128 IC50 = 6600 nM T57392 C0HA4Y 23626131 IC50 > 20000 nM T57392 C3Z6LM 23626132 IC50 > 20000 nM T57392 C2EXB1 23626439 IC50 > 20000 nM T57392 C7EK4A 23626924 IC50 > 20000 nM T57392 CW6OB1 23627212 IC50 > 10000 nM T57392 CWAT04 23630291 IC50 > 10000 nM T57392 CMQ6W7 23630305 IC50 > 10000 nM T57392 CY78MC 23631023 IC50 = 6300 nM T57392 C5V6KM 23631112 IC50 = 90 nM T57392 C0YM5F 23631117 IC50 = 21000 nM T57392 CU1M2C 23631288 IC50 = 150 nM T57392 CQ1M3P 23631387 IC50 = 9600 nM T57392 C4LEI9 23631388 IC50 = 200 nM T57392 CHU29W 23635235 IC50 > 10000 nM T57392 CDL4G9 23645678 IC50 > 200000 nM T57392 C1AQ9P 23647882 IC50 > 30000 nM T57392 CTJ2P1 23647883 IC50 = 8200 nM T57392 CU6E5F 23647884 IC50 = 12000 nM T57392 C6NS9I 23647885 IC50 > 30000 nM T57392 CD9IC3 23647886 IC50 = 30000 nM T57392 CPX95O 23647887 IC50 = 3300 nM T57392 CK9D8P 23647888 IC50 = 5700 nM T57392 CX50BA 23647889 IC50 > 30000 nM T57392 C37JMS 23647890 IC50 = 19000 nM T57392 CJ97BQ 23647892 IC50 > 30000 nM T57392 CXP2G5 23647893 IC50 > 30000 nM T57392 C3JBX4 23647894 IC50 > 30000 nM T57392 C71DGY 23647895 IC50 = 30000 nM T57392 C5LU8P 23647897 IC50 = 6960 nM T57392 C2YVQ3 23647898 IC50 > 30000 nM T57392 C4H5PR 23647899 IC50 > 30000 nM T57392 CW6Y9I 23647900 IC50 = 1890 nM T57392 CMF8R6 23647901 IC50 = 15100 nM T57392 CR7CO9 23647902 IC50 > 30000 nM T57392 CX37CO 23647903 IC50 = 27900 nM T57392 CMG8T2 23647904 IC50 = 3220 nM T57392 C9H7NY 23647905 IC50 = 20600 nM T57392 C3MSV0 23647907 IC50 = 430 nM T57392 CZ0QF1 23648867 IC50 > 30000 nM T57392 CK76FP 23649427 IC50 > 100 nM T57392 CAUC58 23649669 IC50 > 100000 nM T57392 CCL15O 23652787 IC50 = 28800 nM T57392 CKW7V5 23653135 IC50 = 39200 nM T57392 CG39XH 23654666 IC50 > 100 nM T57392 C6VSO8 23657438 IC50 = 5000 nM T57392 CFMX27 23658550 IC50 = 2900 nM T57392 CM7C4W 23661708 IC50 = 20600 nM T57392 CO6L9F 23661716 IC50 = 55400 nM T57392 CHR14F 23661718 IC50 = 8800 nM T57392 C5D3RZ 23683143 IC50 > 50000 nM T57392 C26ANU 23696680 IC50 > 100000 nM T57392 CASU54 23696973 IC50 > 100000 nM T57392 CE4G3V 23729147 IC50 = 9380 nM T57392 CS5E6J 23729988 IC50 > 900000 nM T57392 CK2Q5J 24180592 IC50 > 10000 nM T57392 C9R1PK 24180717 IC50 > 20000 nM T57392 CZ03FI 24649020 IC50 > 50000 nM T57392 CQ35ZB 24743795 IC50 > 50000 nM T57392 C8RC9P 24744325 IC50 > 10000 nM T57392 CSG9V8 24749508 IC50 = 77000 nM T57392 C6JF2R 24753412 IC50 = 49000 nM T57392 CHU49V 24757938 IC50 > 50000 nM T57392 C25HKJ 24758044 IC50 > 40000 nM T57392 CJL67N 24759089 IC50 > 10000 nM T57392 CR9ZI2 24764491 IC50 > 50000 nM T57392 C3P7IS 24768572 IC50 = 35700 nM T57392 CHI83W 24769038 IC50 > 50 nM T57392 C85ELO 24771983 IC50 > 33000 nM T57392 CI7S2G 24782486 IC50 = 50 nM T57392 C6ORA8 24783140 IC50 > 10000 nM T57392 CXSZ08 24783396 IC50 < 50000 nM T57392 CUM03S 24798754 IC50 = 44000 nM T57392 CR48VC 24809711 IC50 = 74000 nM T57392 CY8X0J 24811794 IC50 > 30000 nM T57392 CK02ZF 24812771 IC50 > 50000 nM T57392 C6H2KZ 24817638 IC50 > 30000 nM T57392 C24UQW 24822428 IC50 > 50000 nM T57392 CROH43 24822429 IC50 = 700 nM T57392 C73LOX 24824080 IC50 = 12000 nM T57392 CFI7E9 24824316 IC50 = 17000 nM T57392 CGDB50 24824447 IC50 > 50000 nM T57392 CLU56Y 24824450 IC50 > 50000 nM T57392 CF75DJ 24824494 IC50 = 24000 nM T57392 CLB5M8 24825514 IC50 = 1926 nM T57392 C8DQR0 24825515 IC50 = 1785 nM T57392 C41FJM 24825519 IC50 = 543 nM T57392 CIM1V9 24825522 IC50 = 292 nM T57392 CQN3Z7 24825710 IC50 > 40000 nM T57392 CN4Z2J 24825807 IC50 = 8000 nM T57392 CJ6Z9E 24826945 IC50 = 8000 nM T57392 C1P3IL 24826949 IC50 = 6000 nM T57392 CM2Y0L 24827043 IC50 <= 1000 nM T57392 C2K1OE 24830571 IC50 = 8700 nM T57392 CP9K4V 24834032 IC50 = 60000 nM T57392 CR7X1M 24856034 IC50 > 10000 nM T57392 C61KPI 24856363 IC50 > 10000 nM T57392 CB4LY1 24857598 IC50 > 10000 nM T57392 CSR8J4 24857759 IC50 = 265 nM T57392 CM80JI 24863522 IC50 = 33000 nM T57392 C4UEM5 24871537 IC50 = 1350 nM T57392 CP2L5B 24871655 IC50 = 20 nM T57392 CM8BS1 24879232 IC50 > 5000 nM T57392 CX79IO 24882359 IC50 = 400 nM T57392 CKRF92 24888487 IC50 = 97000 nM T57392 C3AU2O 24888812 Ki = 54.7 nM T57392 C0Z2TG 24889346 IC50 = 39000 nM T57392 CU18OW 24890344 IC50 = 1700 nM T57392 CUZ31Q 24890346 IC50 = 11000 nM T57392 C32TKP 24890348 IC50 = 2200 nM T57392 CU4HV5 24890872 IC50 = 17000 nM T57392 CI53SE 24893978 IC50 = 2200 nM T57392 CNQ6I4 24894028 IC50 > 20000 nM T57392 CDI7N3 24897002 IC50 > 50000 nM T57392 C8GN9W 24899993 IC50 > 50000 nM T57392 CZSA05 24899995 IC50 > 50000 nM T57392 CIZ6O1 24900235 IC50 > 50000 nM T57392 C61ARF 24900236 IC50 > 50000 nM T57392 C7J4ZQ 24900259 IC50 > 40000 nM T57392 CUY89J 24936155 Ki = 15000 nM T57392 CC4K1P 24949545 IC50 = 6300 nM T57392 C17QKF 24949548 IC50 = 18000 nM T57392 CCA9G2 24949700 IC50 = 16000 nM T57392 CFU0T1 24949702 IC50 = 66000 nM T57392 CE79PI 24949704 IC50 = 25000 nM T57392 CI7NG8 24951587 IC50 > 8000 nM T57392 CLZ23U 24951610 IC50 > 30000 nM T57392 CNP3T1 24951733 IC50 = 16000 nM T57392 CEGV39 24951942 IC50 > 10000 nM T57392 C9EH3S 24951943 IC50 > 10000 nM T57392 CW9UN1 24951944 IC50 > 10000 nM T57392 CP98YL 24951946 IC50 > 10000 nM T57392 C3VO7Q 24960588 IC50 = 100000 nM T57392 CZ89IP 24961687 IC50 = 34000 nM T57392 CW4X0E 24962988 IC50 = 1210 nM T57392 CB68JF 24963286 IC50 = 3600 nM T57392 C5EIW1 24965329 IC50 = 16800 nM T57392 C6U2AP 24965679 IC50 = 19500 nM T57392 CM6I1G 24967634 IC50 = 1400 nM T57392 C0XS2D 24967990 IC50 = 1600 nM T57392 C71CNA 24967991 IC50 = 25100 nM T57392 CT39VO 24969452 IC50 = 740 nM T57392 CGZ60N 24969453 IC50 = 250 nM T57392 CE95WV 24970356 IC50 = 22900 nM T57392 CF0A5P 24984572 IC50 > 10000 nM T57392 CQ2Z7T 24985115 IC50 > 10000 nM T57392 CM7HQ5 24985395 IC50 > 20000 nM T57392 CEJ74C 24985745 IC50 > 20000 nM T57392 C27WVS 24986404 IC50 > 100000 nM T57392 C94AHE 24988956 IC50 > 100000 nM T57392 C14EFU 24990122 IC50 = 6700 nM T57392 C80LEK 24990485 IC50 = 19000 nM T57392 CMD98H 24990837 IC50 > 33000 nM T57392 CNMD47 24990839 IC50 = 20000 nM T57392 C0I5NG 24991884 IC50 > 100000 nM T57392 CL83OS 24992519 IC50 > 30000 nM T57392 CK0NZ8 24993163 IC50 > 10000 nM T57392 C8KIP6 24993178 IC50 > 30000 nM T57392 CD8U2B 24993500 IC50 > 30000 nM T57392 CCDF20 24994127 IC50 > 11000 nM T57392 CDF57P 24995525 IC50 = 5011.87 nM T57392 CJM8R0 24996322 IC50 > 30000 nM T57392 C2BPD5 25005270 IC50 > 50000 nM T57392 CT64BR 25005273 IC50 = 34000 nM T57392 CX0O4A 25005628 IC50 = 21000 nM T57392 CR9LQ8 25005629 IC50 = 23000 nM T57392 CWBO80 25005631 IC50 = 19000 nM T57392 C8ZQ3E 25005985 IC50 = 10000 nM T57392 C47CFM 25005986 IC50 = 10000 nM T57392 CKT5V7 25005987 IC50 = 10000 nM T57392 C5NF9P 25005988 IC50 = 19000 nM T57392 C2H8XF 25005989 IC50 > 25000 nM T57392 C1MWK0 25005990 IC50 > 50000 nM T57392 CX3I6O 25008509 IC50 > 10000 nM T57392 C0C3ZJ 25008854 IC50 > 10000 nM T57392 CX8N1E 25009027 IC50 > 10000 nM T57392 C30HJO 25009028 IC50 > 10000 nM T57392 C3C6HW 25009031 IC50 > 10000 nM T57392 CZ6T5Q 25009937 IC50 > 29000 nM T57392 CU7G9E 25010550 IC50 < 10000 nM T57392 C32AUW 25013308 IC50 > 10000 nM T57392 C1VRJ3 25014630 IC50 = 750 nM T57392 CP13LW 25016311 IC50 = 27000 nM T57392 C91QFN 25019282 IC50 = 180000 nM T57392 CMU30E 25022640 IC50 > 100000 nM T57392 CQ9LS6 25022704 IC50 = 3400 nM T57392 CF67EB 25023856 IC50 = 10000 nM T57392 C0L9PQ 25023857 IC50 < 10000 nM T57392 CA2T1X 25023858 IC50 < 10000 nM T57392 C7SKU1 25023859 IC50 < 10000 nM T57392 CA20NZ 25025581 IC50 = 4000 nM T57392 CPJD86 25025779 IC50 > 4000 nM T57392 CDX2C6 25025977 IC50 > 8000 nM T57392 C0LO9C 25028373 IC50 = 100000 nM T57392 CKLQ76 25028375 IC50 = 54000 nM T57392 CDKJ78 25033361 IC50 > 40000 nM T57392 CXDF80 25034348 IC50 > 200000 nM T57392 CR3I9Y 25050394 EC50 > 100000 nM T57392 C86CQY 25052759 IC50 < 500 nM T57392 CVQS96 25052767 IC50 > 25000 nM T57392 CZO27W 25054032 IC50 > 30000 nM T57392 C7EQ5T 25054288 IC50 > 10000 nM T57392 CN2G3K 25054307 IC50 > 30000 nM T57392 C7EXD5 25054568 IC50 > 30000 nM T57392 C1PKF0 25056080 IC50 > 10000 nM T57392 CFHO90 25056112 IC50 > 30000 nM T57392 C6Z3CE 25057124 IC50 > 10000 nM T57392 CH6AU8 25057408 IC50 > 30000 nM T57392 C0B7RT 25057409 IC50 > 30000 nM T57392 C3AT0H 25057667 IC50 > 30000 nM T57392 CH7YC4 25057933 IC50 > 30000 nM T57392 CPT9X8 25066443 IC50 > 10000 nM T57392 CA76KJ 25067046 IC50 = 800 nM T57392 CGMN97 25067404 IC50 = 24000 nM T57392 CMJ1F7 25067546 IC50 = 600 nM T57392 C7YRG0 25067560 IC50 = 7.943 nM T57392 CMH41V 25069448 IC50 = 24800 nM T57392 CBY3O2 25070582 IC50 > 30000 nM T57392 CP9J7Q 25071019 IC50 = 220 nM T57392 CBRM65 25074167 IC50 = 40000 nM T57392 C1AGW7 25093241 IC50 = 2100 nM T57392 CH90KV 25097876 IC50 > 10000 nM T57392 CAO38V 25098429 IC50 > 10000 nM T57392 CF7ON5 25099235 IC50 > 50000 nM T57392 CUYI02 25101821 IC50 > 10000 nM T57392 CP7MH1 25106114 IC50 < 500 nM T57392 C98CGM 25106115 IC50 < 500 nM T57392 CLD7X0 25107258 IC50 < 500 nM T57392 C4NE6H 25107259 IC50 < 500 nM T57392 COT5G4 25107260 IC50 < 500 nM T57392 C0K9HA 25110600 IC50 > 14000 nM T57392 CKRN07 25118654 IC50 > 50000 nM T57392 CZ96TL 25118804 IC50 = 2000 nM T57392 C8T7NC 25118805 IC50 > 50000 nM T57392 CNT2S6 25119161 IC50 = 1100 nM T57392 C29RAS 25119164 IC50 = 2200 nM T57392 C3GI7J 25119513 IC50 = 1800 nM T57392 CT67MA 25119856 IC50 = 1300 nM T57392 C3UW6I 25119857 IC50 = 390 nM T57392 CR0CZ5 25119860 IC50 < 780 nM T57392 CDO26T 25129042 IC50 > 31622.78 nM T57392 C9Z6UG 25138295 IC50 = 100000 nM T57392 CHS25Z 25141776 IC50 > 5000 nM T57392 CE93TF 25141777 IC50 > 5000 nM T57392 C1AIH7 25141896 IC50 > 5000 nM T57392 CWF5Z3 25143506 IC50 > 30000 nM T57392 CFS3N9 25144422 IC50 > 20000 nM T57392 C78YWA 25145716 IC50 > 20000 nM T57392 C35XQI 25150621 IC50 = 6000 nM T57392 CAVR45 25150711 IC50 = 6000 nM T57392 CL1W5D 25154436 IC50 > 10000 nM T57392 C67QXP 25154827 IC50 = 13300 nM T57392 C8AC0Y 25154864 IC50 = 3900 nM T57392 CGH08V 25164128 IC50 = 15000 nM T57392 C3NVW5 25165471 IC50 > 15000 nM T57392 CF9KY4 25165474 IC50 > 15000 nM T57392 CW9MX8 25168440 IC50 = 4100 nM T57392 CXC35U 25168857 IC50 = 800 nM T57392 CH06WV 25168930 IC50 > 10000 nM T57392 C5TJD2 25172265 IC50 > 10000 nM T57392 CJMZ37 25174150 IC50 > 7500 nM T57392 C0XHA2 25180109 IC50 < 200000 nM T57392 C90UKD 25180304 IC50 < 200000 nM T57392 C6ZE9H 25180500 IC50 < 200000 nM T57392 CK6Z9J 25181419 IC50 > 100000 nM T57392 CGE8V0 25181656 IC50 > 20000 nM T57392 CZUP40 25181801 IC50 > 20000 nM T57392 C5AKX1 25181802 IC50 > 20000 nM T57392 C6EWF1 25183622 IC50 > 30000 nM T57392 C79LPB 25183668 IC50 > 20000 nM T57392 CHJY51 25183669 IC50 > 2000 nM T57392 C0Q8BN 25183817 IC50 > 20000 nM T57392 CF46YL 25183819 IC50 > 20000 nM T57392 C89CXW 25183820 IC50 > 20000 nM T57392 C5C7GH 25184832 IC50 > 10000 nM T57392 CSU0B5 25189891 IC50 > 15000 nM T57392 C04QGB 25190493 IC50 > 89000 nM T57392 CV3TA6 25192021 IC50 > 7500 nM T57392 C9UL8Y 25192468 IC50 > 7500 nM T57392 C7A8UE 25192471 IC50 > 7500 nM T57392 CH3L6V 25192656 IC50 > 10000 nM T57392 C46ANM 25195291 IC50 = 10600 nM T57392 C8CY6O 25205318 IC50 > 10000000 nM T57392 CY1M9Q 25205319 IC50 > 10000000 nM T57392 CLFM35 25206064 IC50 > 10000 nM T57392 CTBK98 25208406 Ki = 28.1 nM T57392 C37YTG 25210603 IC50 > 10000 nM T57392 CW3JR1 25210604 IC50 = 300 nM T57392 CTQM87 25210756 IC50 > 25000 nM T57392 CE7BA0 25210873 IC50 = 1000 nM T57392 C0FE8U 25210874 IC50 < 100 nM T57392 C2UQJ6 25211598 EC50 > 100000 nM T57392 CKI86X 25211805 EC50 > 100000 nM T57392 CHW2X0 25211910 EC50 > 100000 nM T57392 CXH7F8 25218692 IC50 = 1600 nM T57392 CUN19O 25218744 IC50 > 20000 nM T57392 CE40LR 25222164 IC50 = 8300 nM T57392 CJ65AE 25226377 IC50 > 50000 nM T57392 CIZB04 25254173 IC50 = 14000 nM T57392 CW9JM2 25256832 IC50 > 10000 nM T57392 C3GC7P 25256833 IC50 > 10000 nM T57392 CI8SQ7 25263541 IC50 = 20000 nM T57392 CTW7E8 25263542 IC50 > 20000 nM T57392 C6DX5M 25264621 IC50 < 80 nM T57392 C32USM 25264907 IC50 < 80 nM T57392 CJ50IN 25265057 IC50 = 80 nM T57392 C20XDK 25265635 IC50 > 20000 nM T57392 CJ32HC 25265835 IC50 > 25000 nM T57392 CGQ8D3 25270849 IC50 = 22700 nM T57392 CI1G2C 26873419 IC50 = 19900 nM T57392 C7PK2X 29938807 IC50 > 20000 nM T57392 C0FA2X 40680501 IC50 = 2630 nM T57392 CE63OB 40700807 IC50 = 1300 nM T57392 CHW3D1 40700815 IC50 = 10600 nM T57392 CBH1P0 42210730 IC50 > 30000 nM T57392 CT0NF6 42415086 IC50 = 6700 nM T57392 CKH3P1 42606928 IC50 > 40000 nM T57392 C1YO7H 42618040 EC50 > 100000 nM T57392 CN34WV 42618054 EC50 > 100000 nM T57392 C0I4MK 42618066 EC50 > 100000 nM T57392 CGU3N8 42618068 EC50 = 21000 nM T57392 CY4LG8 42622934 IC50 > 75000 nM T57392 CJ8LY0 42626024 IC50 = 11000 nM T57392 CS04KE 42629368 IC50 > 20000 nM T57392 CYGN52 42629369 IC50 > 20000 nM T57392 C3LK1F 42637004 IC50 > 10000 nM T57392 CRA13T 42637062 IC50 = 3960 nM T57392 C7PHI5 42637065 IC50 = 3730 nM T57392 CI29GP 42637133 IC50 = 1300 nM T57392 C6NAD9 42637280 IC50 = 20000 nM T57392 C7JX9R 42637281 IC50 > 10000 nM T57392 CR2HI3 42637282 IC50 = 1320 nM T57392 C4MON9 42637355 IC50 = 4270 nM T57392 C78OHW 42637357 IC50 = 1000 nM T57392 CAN25J 42637358 IC50 = 2900 nM T57392 CL98FP 42637359 IC50 > 10000 nM T57392 CT6G1Z 42637431 IC50 = 3300 nM T57392 CF1ZC7 42637498 IC50 > 10000 nM T57392 CCH5J9 42637980 IC50 > 10000 nM T57392 CBO9N2 42637982 IC50 = 20000 nM T57392 CY0WG9 42638063 IC50 = 13000 nM T57392 CH3MY1 42639933 IC50 = 4100 nM T57392 CVY8H2 42640092 IC50 = 13000 nM T57392 C4P1IM 42643589 IC50 < 10000 nM T57392 CX9SM6 42643591 IC50 = 10000 nM T57392 C96FIN 42644084 IC50 > 10000 nM T57392 C8BI5F 42644088 IC50 > 10000 nM T57392 CREJ31 42646199 IC50 > 10000 nM T57392 CKZ76R 42646202 IC50 > 10000 nM T57392 C81NVM 42646450 IC50 > 10000 nM T57392 CVBO78 42647178 IC50 < 10000 nM T57392 C2MY8X 42647277 IC50 < 200 nM T57392 CZF5G9 42916879 IC50 > 10000 nM T57392 C5E6UL 43388611 IC50 = 4170 nM T57392 CS40ML 44123747 IC50 = 38000 nM T57392 CS0H1B 44125704 IC50 > 50000 nM T57392 C47OXT 44128987 IC50 > 50000 nM T57392 CN5O1Y 44129065 IC50 > 50000 nM T57392 CX7W2E 44132009 IC50 = 65000 nM T57392 CXS43I 44132271 IC50 = 900 nM T57392 CA7HI4 44137226 IC50 > 10000 nM T57392 C5O1MR 44137674 IC50 > 10000 nM T57392 CG73ST 44138103 IC50 > 30000 nM T57392 C6QY9W 44143257 IC50 = 11000 nM T57392 C3RKI7 44158698 IC50 = 1700 nM T57392 CO60AP 44159044 IC50 = 1000 nM T57392 C5G4LN 44159411 IC50 > 30000 nM T57392 CHI65U 44159530 IC50 > 30000 nM T57392 C9RC2Z 44159640 IC50 = 600 nM T57392 C1C2DH 44159759 IC50 = 700 nM T57392 CMNH53 44159772 IC50 > 30000 nM T57392 C5GYS4 44160248 IC50 > 50000 nM T57392 C25DHI 44178203 IC50 = 220 nM T57392 CPF50A 44184875 IC50 > 24000 nM T57392 CH7FJ6 44188689 IC50 = 580 nM T57392 CSE8X3 44188690 IC50 = 1900 nM T57392 CY2Q9O 44188691 IC50 = 350 nM T57392 C6FPM5 44188693 IC50 = 40 nM T57392 CWR04I 44188695 IC50 = 310 nM T57392 CJEG24 44188861 IC50 = 300 nM T57392 C9XSI6 44189029 IC50 = 700 nM T57392 C2XE7Y 44189733 IC50 = 16000 nM T57392 CSN2I3 44190675 IC50 = 7000 nM T57392 CA9FN6 44193857 IC50 < 500 nM T57392 CE5A9Z 44193858 IC50 < 500 nM T57392 CFEX37 44193859 IC50 < 500 nM T57392 CBC3W9 44193860 IC50 < 500 nM T57392 C19RXP 44193960 IC50 < 500 nM T57392 CEM1J3 44193962 IC50 < 500 nM T57392 CU06VM 44193963 IC50 < 500 nM T57392 CE1PW4 44194155 IC50 < 500 nM T57392 C5L6WO 44194849 IC50 > 10000 nM T57392 CBS1D6 44195184 IC50 < 500 nM T57392 C5T3FW 44195186 IC50 < 200 nM T57392 CZ29JY 44205724 IC50 > 30000 nM T57392 C5RL9M 44215838 IC50 = 3700 nM T57392 C2KJB0 44216880 IC50 = 100 nM T57392 C7VWX5 44220300 IC50 > 10000 nM T57392 C2O0NL 44230575 IC50 > 20000 nM T57392 CA46YO 44230734 IC50 = 100 nM T57392 CB5P7N 44230873 IC50 = 3500 nM T57392 CXI7Z8 44230875 IC50 = 300 nM T57392 CU8MS7 44230877 IC50 = 800 nM T57392 C67PRE 44231009 IC50 = 2600 nM T57392 C67WIP 44231010 IC50 = 8700 nM T57392 CCP13S 44231144 IC50 = 400 nM T57392 CIBR82 44231149 IC50 = 4800 nM T57392 CE12BT 44231265 IC50 = 2900 nM T57392 C0TF4H 44231266 IC50 = 600 nM T57392 C7HCZ5 44231267 IC50 = 7500 nM T57392 CDZ8F4 44231268 IC50 = 11500 nM T57392 CX4YL8 44232522 IC50 > 10000 nM T57392 CQ13MH 44234032 IC50 > 50000 nM T57392 C7UY5F 44235863 IC50 > 10000 nM T57392 CX2W8Y 44236320 IC50 > 10000 nM T57392 C8LN0U 44236321 IC50 > 10000 nM T57392 CK4S5Y 44236322 IC50 < 10000 nM T57392 CF8HE4 44245734 IC50 = 7200 nM T57392 C4W0SH 44247585 IC50 > 40000 nM T57392 CH59RP 44247803 IC50 = 300 nM T57392 C7MY2N 44247806 IC50 = 50000 nM T57392 CF9TE1 44247935 IC50 = 3300 nM T57392 CDOA12 44249906 IC50 > 41000 nM T57392 C85DHY 44250284 IC50 = 11000 nM T57392 C8P2LE 44250288 IC50 > 10000 nM T57392 CLY1A3 44251218 IC50 > 25000 nM T57392 C1O8LH 44253973 IC50 = 2200 nM T57392 C47RZO 44254057 IC50 = 7100 nM T57392 C41MNG 44254058 IC50 = 2100 nM T57392 C2SVL6 44254059 IC50 = 640 nM T57392 CVW13I 44254060 IC50 = 5700 nM T57392 C0NZW8 44254061 IC50 = 33000 nM T57392 C3N2KB 44254062 IC50 = 9500 nM T57392 CJW3P2 44254063 IC50 = 4600 nM T57392 C6OJS0 44254504 IC50 = 670 nM T57392 CSBD48 44254505 IC50 = 2800 nM T57392 C1IPQ6 44254506 IC50 = 4700 nM T57392 CTL57U 44254584 IC50 = 7600 nM T57392 CZY2S1 44254585 IC50 = 1000 nM T57392 C9SQ8D 44254859 IC50 = 1200 nM T57392 CB47EJ 44254954 IC50 = 4100 nM T57392 C79QBX 44254955 IC50 = 4400 nM T57392 CVCP62 44254956 IC50 = 1800 nM T57392 CK7B1Q 44254957 IC50 = 2800 nM T57392 CJH6K5 44255041 IC50 = 2400 nM T57392 C5Z9KH 44255042 IC50 = 3100 nM T57392 C1FE8D 44255043 IC50 = 21000 nM T57392 CGB3A7 44255044 IC50 = 5300 nM T57392 CTY9U6 44255045 IC50 = 7500 nM T57392 CNO97U 44255810 IC50 = 18000 nM T57392 C4XW9G 44266800 IC50 = 47000 nM T57392 C0NFL2 44269753 Ki = 3200 nM T57392 C23SRP 44269789 Ki = 9700 nM T57392 C1U8OW 44269925 Ki = 1100 nM T57392 CB9L7J 44289715 IC50 = 14000 nM T57392 C6UR1Q 44289919 IC50 = 37700 nM T57392 CMUT04 44289926 IC50 = 2200 nM T57392 CQ4Y0G 44289927 IC50 = 1600 nM T57392 CHM25N 44290039 IC50 = 500 nM T57392 C8DF0N 44303648 Ki = 2000 nM T57392 C5PJ2E 44303662 Ki = 3000 nM T57392 CGI67V 44303681 Ki = 1000 nM T57392 CU23OI 44303706 Ki = 100 nM T57392 C1R9SH 44303742 Ki = 600 nM T57392 CYX1H6 44303755 Ki = 700 nM T57392 CNTG98 44303756 Ki = 1000 nM T57392 CV5B4U 44303960 Ki = 2000 nM T57392 CDJ7N5 44303965 Ki = 8000 nM T57392 C3K2YT 44303992 Ki = 5000 nM T57392 CFH86V 44303993 Ki = 4000 nM T57392 CU9V4N 44304000 Ki = 10000 nM T57392 C0Z7SV 44304001 Ki = 30000 nM T57392 C9L0UY 44304110 Ki = 3000 nM T57392 CYQ5B9 44304132 Ki = 5000 nM T57392 CFT97O 44304149 Ki = 3000 nM T57392 CV8JB7 44304166 Ki = 10000 nM T57392 CKM9U8 44304170 Ki = 7000 nM T57392 CRW21Q 44304185 Ki = 2000 nM T57392 CLJ62O 44304196 Ki = 4000 nM T57392 CTC9F0 44304204 Ki = 1000 nM T57392 C6BK8U 44304206 Ki = 4000 nM T57392 CTHB52 44304210 Ki = 8000 nM T57392 C3HS5O 44304365 Ki = 2000 nM T57392 CD9TP4 44304366 Ki = 2000 nM T57392 CLV8R6 44304367 Ki = 1000 nM T57392 CN6O1V 44304368 Ki = 4000 nM T57392 CZE1S8 44304386 Ki = 3000 nM T57392 CP5D6R 44304434 Ki = 7000 nM T57392 CF4UC9 44304435 Ki = 3000 nM T57392 C7S2ZI 44340870 IC50 = 3200 nM T57392 CE13FX 44341241 IC50 = 1050 nM T57392 CX65PH 44341461 IC50 = 400 nM T57392 C0KD4U 44346053 IC50 > 2000 nM T57392 CH0O5Q 44346322 IC50 > 2000 nM T57392 C5OQ2K 44366980 IC50 > 100000 nM T57392 CM6V4C 44388606 IC50 = 217000 nM T57392 CKV1H9 44388612 IC50 = 297000 nM T57392 CGU79D 44388657 IC50 = 197000 nM T57392 CMV75Q 44389639 IC50 = 21000 nM T57392 C62EIF 44389641 IC50 = 50 nM T57392 CW1C0L 44389644 IC50 = 100000 nM T57392 C92ACP 44389656 IC50 = 420 nM T57392 CPM6Z1 44389661 IC50 = 3800 nM T57392 C7P3EL 44389686 IC50 = 12000 nM T57392 C8E9GR 44389691 IC50 = 120 nM T57392 C5U1ZL 44389692 IC50 = 4800 nM T57392 CPX96I 44389701 IC50 = 280 nM T57392 CN3C0B 44389708 IC50 = 2100 nM T57392 CE6A3T 44389759 IC50 = 50 nM T57392 C8FCN7 44389771 IC50 = 350 nM T57392 CV9QW5 44389774 IC50 = 40 nM T57392 CN3M9I 44389788 IC50 = 110 nM T57392 CY7T0R 44389831 IC50 = 70 nM T57392 C07TLH 44389866 IC50 = 90 nM T57392 C7FN0P 44389886 IC50 = 670 nM T57392 C0IG4E 44389899 IC50 = 40 nM T57392 C02ONK 44389924 IC50 = 30 nM T57392 CQJ8B1 44389927 IC50 = 40 nM T57392 CUJ27R 44389944 IC50 = 120 nM T57392 C80BAX 44396806 IC50 = 310000 nM T57392 CRL7Y5 44399273 IC50 = 326 nM T57392 C56JOK 44399274 IC50 = 35 nM T57392 C3M4XI 44399378 IC50 = 18 nM T57392 CPSF28 44399379 IC50 = 107 nM T57392 C1NX9P 44399492 IC50 = 600 nM T57392 CC1UY9 44399493 IC50 = 5702 nM T57392 C4XEQ2 44399584 IC50 = 295 nM T57392 CR0G7H 44399648 IC50 = 4776 nM T57392 CT2YO6 44399674 IC50 = 1820 nM T57392 CMA91N 44399675 IC50 = 1037 nM T57392 C9GF1J 44399730 IC50 = 1220 nM T57392 CUGE51 44403300 IC50 = 23000 nM T57392 CE41AD 44405138 IC50 = 6200 nM T57392 CN0G4K 44405139 IC50 = 150 nM T57392 CU02RP 44405141 IC50 = 770 nM T57392 CUIG59 44405142 IC50 = 14000 nM T57392 CA2B3X 44405144 IC50 = 1600 nM T57392 C1UZE3 44405145 IC50 = 2900 nM T57392 CYX81F 44405161 IC50 = 320 nM T57392 C14OGA 44405162 IC50 = 6700 nM T57392 CHU8N9 44405164 IC50 = 9500 nM T57392 C0AXJ5 44405165 IC50 = 11 nM T57392 CV5Y3I 44405172 IC50 = 7400 nM T57392 C32CVQ 44405173 IC50 = 1800 nM T57392 CE43NQ 44405175 IC50 = 4800 nM T57392 CZI0A4 44405840 IC50 = 0.1 nM T57392 CZG7V0 44407893 IC50 = 300 nM T57392 C54DYN 44407894 IC50 = 2000 nM T57392 C0NT5I 44407898 IC50 = 1000 nM T57392 C1J5QH 44407899 IC50 > 20000 nM T57392 CL17UJ 44407912 IC50 = 1000 nM T57392 C6YX7H 44407913 IC50 = 3000 nM T57392 CF76BI 44407936 IC50 > 30000 nM T57392 C24JPG 44407943 IC50 = 900 nM T57392 CK09NT 44407949 IC50 = 30000 nM T57392 CL6I5U 44407954 IC50 = 3000 nM T57392 C07FOH 44407955 IC50 = 2000 nM T57392 C4MD9V 44407992 IC50 = 6000 nM T57392 CA52BY 44408005 IC50 > 30000 nM T57392 CQF0X2 44408010 IC50 = 2000 nM T57392 C78PQK 44408011 IC50 = 12000 nM T57392 C7UW4T 44408015 IC50 = 2000 nM T57392 C3IA8O 44408021 IC50 = 3000 nM T57392 C9Z6EP 44408029 IC50 > 20000 nM T57392 C9I6CN 44408030 IC50 = 3000 nM T57392 CY89AT 44408034 IC50 > 30000 nM T57392 CNK39Z 44408035 IC50 > 30000 nM T57392 CHZ1T2 44408036 IC50 = 1000 nM T57392 CWD6E7 44408037 IC50 > 20000 nM T57392 C3WRS0 44408041 IC50 = 4000 nM T57392 CSKW61 44408042 IC50 = 6000 nM T57392 CG4A3D 44408054 IC50 = 300 nM T57392 CZ2R5C 44408055 IC50 = 2000 nM T57392 C87TDO 44408063 IC50 = 9000 nM T57392 CS4UZ8 44408110 IC50 = 6000 nM T57392 CK4A6E 44408116 IC50 = 6000 nM T57392 CH2V3I 44408118 IC50 = 5000 nM T57392 CP53NT 44409473 IC50 = 5800 nM T57392 CA3B0O 44409475 IC50 > 200000 nM T57392 C05WIJ 44409476 IC50 = 40000 nM T57392 CCH84T 44409480 IC50 = 60000 nM T57392 C0PO6W 44409488 IC50 > 400000 nM T57392 C0SXD3 44410799 IC50 > 5000 nM T57392 CR4HX5 44410840 IC50 > 5000 nM T57392 C73OZJ 44410841 IC50 > 5000 nM T57392 C7E4LF 44413712 IC50 > 30000 nM T57392 CO2M8L 44413775 IC50 = 9000 nM T57392 CP5G8I 44413790 IC50 > 30000 nM T57392 CQD2S5 44414696 IC50 = 3600 nM T57392 CF8Q6Y 44414836 IC50 = 10000 nM T57392 CMV57G 44415389 IC50 = 55 nM T57392 C0OG4J 44415524 IC50 = 3300 nM T57392 C7JV9E 44416651 IC50 = 3162.28 nM T57392 C8ZI4H 44416671 IC50 = 5011.87 nM T57392 CJ08ZR 44416753 IC50 = 2300 nM T57392 C3O7GK 44416757 IC50 = 3981.07 nM T57392 CY6T2S 44416782 IC50 > 30000 nM T57392 C0SX4T 44416786 IC50 = 24500 nM T57392 C9R1UT 44416800 IC50 = 2511.89 nM T57392 CMHX86 44416801 IC50 > 10000 nM T57392 C4W8ST 44416859 IC50 = 3981.07 nM T57392 CG46MT 44416862 IC50 = 18700 nM T57392 CT62LG 44416877 IC50 = 4500 nM T57392 C8ELH9 44416880 IC50 > 30000 nM T57392 C76SRF 44416881 IC50 = 5011.87 nM T57392 CDNH81 44416895 IC50 = 900 nM T57392 C2FX5H 44416898 IC50 > 30000 nM T57392 CLP16U 44416911 IC50 = 3500 nM T57392 C0X5HE 44416916 IC50 > 30000 nM T57392 C7BI9T 44416969 IC50 = 9200 nM T57392 CIEB89 44416970 IC50 = 15600 nM T57392 C9QU0R 44416989 IC50 = 6309.57 nM T57392 C8BQ3P 44416990 IC50 > 30000 nM T57392 C05LZR 44417024 IC50 > 30000 nM T57392 CZ5SQ3 44417025 IC50 > 30000 nM T57392 C0A2FS 44417069 IC50 = 12500 nM T57392 CQ2D0O 44418482 IC50 > 25000 nM T57392 CX09NV 44418490 IC50 = 7000 nM T57392 CY2F3Q 44420235 IC50 > 10000 nM T57392 CH1R7M 44420600 IC50 > 10000 nM T57392 CU52GB 44425701 IC50 = 1600 nM T57392 CX8TR0 44425719 IC50 = 19000 nM T57392 CV7N0H 44425963 IC50 = 5100 nM T57392 C7G6VX 44426995 Ki = 5000 nM T57392 CAWL05 44428924 IC50 > 100000 nM T57392 CODL74 44430453 IC50 = 8600 nM T57392 CNW86X 44430460 IC50 = 3400 nM T57392 CJ9C8U 44430475 IC50 = 22500 nM T57392 CTB82G 44431744 IC50 > 50000 nM T57392 CL6B7S 44431775 IC50 = 11000 nM T57392 CQC0U9 44433394 Ki = 840 nM T57392 C9LM7U 44433789 IC50 = 24000 nM T57392 CWDJ93 44433797 IC50 = 92000 nM T57392 CU67NA 44433798 IC50 = 57000 nM T57392 CNU4B6 44433799 IC50 = 73000 nM T57392 C5V7WE 44433800 IC50 > 100000 nM T57392 CBP25Q 44433802 IC50 > 100000 nM T57392 CB1SD9 44433803 IC50 = 63000 nM T57392 CP2G6L 44440493 IC50 = 4700 nM T57392 CXSQ75 44440525 IC50 > 30000 nM T57392 C2VAG9 44440645 IC50 = 98 nM T57392 C08ZST 44440659 IC50 > 10000 nM T57392 CR3PM7 44440662 IC50 > 10000 nM T57392 CCSI57 44440665 IC50 > 10000 nM T57392 CDEY23 44441334 IC50 = 30 nM T57392 COBN96 44441335 IC50 = 500 nM T57392 C23BGW 44441336 IC50 = 100 nM T57392 CJ2S0W 44441340 IC50 = 9400 nM T57392 C1R0DN 44441341 IC50 = 5900 nM T57392 C9FB6Y 44441345 IC50 = 15700 nM T57392 C2GAV7 44441348 IC50 = 5500 nM T57392 CWH92R 44441349 IC50 = 8200 nM T57392 C61VKY 44441350 IC50 = 30000 nM T57392 CF4A8D 44441351 IC50 = 30000 nM T57392 CD30KT 44441353 IC50 = 6800 nM T57392 CKJ62V 44442476 IC50 < 300 nM T57392 CFSZ45 44442477 IC50 = 3900 nM T57392 C6ZK7X 44442478 IC50 = 3500 nM T57392 C9HEW7 44442480 IC50 = 8400 nM T57392 C2X7NQ 44442481 IC50 = 11000 nM T57392 CAC7V9 44442482 IC50 > 30000 nM T57392 CVO5Z2 44442483 IC50 > 30000 nM T57392 CJPR25 44442484 IC50 > 30000 nM T57392 C9NMQ3 44442485 IC50 > 30000 nM T57392 CT0C4I 44443093 IC50 > 20000 nM T57392 CF1V8O 44443098 IC50 = 15000 nM T57392 CHZ48Q 44443101 IC50 = 14000 nM T57392 CQ53TV 44443130 IC50 > 19000 nM T57392 CEZ6U8 44443131 IC50 > 16000 nM T57392 CN4XZ6 44443132 IC50 > 9000 nM T57392 CV5CK0 44443532 IC50 = 7970 nM T57392 CWE9P2 44445839 IC50 = 100 nM T57392 CH7W8P 44445840 IC50 = 490 nM T57392 CY2KD0 44445842 IC50 = 440 nM T57392 C5W8MO 44445843 IC50 = 570 nM T57392 C5OYU7 44445845 IC50 = 20000 nM T57392 C81EKO 44445846 IC50 = 160 nM T57392 CY7XD2 44445847 IC50 = 56000 nM T57392 CRV2Y7 44445849 IC50 = 800 nM T57392 CSC7N1 44445850 IC50 = 28000 nM T57392 CP57AC 44445851 IC50 = 1400 nM T57392 CV6A2C 44445853 IC50 > 100000 nM T57392 C6C1DS 44445854 IC50 = 2100 nM T57392 CY0JI9 44445855 IC50 = 340 nM T57392 CLB89R 44445856 IC50 = 50 nM T57392 C53WTR 44445859 IC50 = 10 nM T57392 C1BVA3 44445861 IC50 = 140 nM T57392 C2BX1W 44445862 IC50 = 60 nM T57392 CQRN92 44445863 IC50 = 1200 nM T57392 C4SA7D 44445864 IC50 = 170 nM T57392 CFZ8R7 44445865 IC50 = 550 nM T57392 COXK37 44445866 IC50 = 5100 nM T57392 COK20T 44445867 IC50 = 2000 nM T57392 CHX93V 44445868 IC50 = 780 nM T57392 CNM14B 44445870 IC50 = 28000 nM T57392 C05MCY 44445872 IC50 = 4300 nM T57392 C8X3DF 44445873 IC50 = 2800 nM T57392 C76VUI 44445874 IC50 = 920 nM T57392 CXH5Z0 44445875 IC50 = 23000 nM T57392 C5P6QX 44445876 IC50 = 2200 nM T57392 CB75CU 44445877 IC50 = 910 nM T57392 C8CKU0 44445878 IC50 = 810 nM T57392 C97UQC 44445879 IC50 = 80 nM T57392 CJFW14 44445880 IC50 = 1500 nM T57392 CUC7P1 44445883 IC50 = 80 nM T57392 C1X3MD 44445884 IC50 = 1200 nM T57392 CCHB32 44445885 IC50 = 1100 nM T57392 CWB3K5 44445886 IC50 = 1200 nM T57392 C56YMC 44445887 IC50 = 500 nM T57392 C7PN6T 44445888 IC50 = 410 nM T57392 CS4XV5 44445889 IC50 = 170 nM T57392 CY2VI3 44445890 IC50 = 3900 nM T57392 COF4U0 44445891 IC50 = 3300 nM T57392 C1H8YR 44445892 IC50 = 740 nM T57392 C3C4DJ 44445893 IC50 = 2200 nM T57392 CWZA43 44445894 IC50 = 1100 nM T57392 C7XL0J 44445895 IC50 = 12000 nM T57392 C3RZY0 44445896 IC50 = 12000 nM T57392 C30QBA 44445901 IC50 = 7400 nM T57392 C01JRH 44445907 IC50 = 680 nM T57392 CR19SE 44445915 IC50 = 1200 nM T57392 C61XVE 44445916 IC50 = 1800 nM T57392 CAOB06 44448056 IC50 = 50 nM T57392 CY8RO4 44448772 IC50 = 2300 nM T57392 C9K8EN 44448775 IC50 = 750 nM T57392 CW7BG9 44448874 IC50 = 8000 nM T57392 CR6TO5 44448876 IC50 = 1700 nM T57392 CF40AD 44448913 IC50 = 3500 nM T57392 C5OR0Q 44448947 IC50 = 2200 nM T57392 C15VTJ 44448976 IC50 = 6700 nM T57392 C1F2MP 44449004 IC50 = 8400 nM T57392 CL9M2D 44449052 IC50 = 21000 nM T57392 CL4H8Y 44449053 IC50 = 2900 nM T57392 C3L4XD 44449079 IC50 = 5100 nM T57392 C4T1MQ 44449106 IC50 = 1600 nM T57392 C9XZY1 44449107 IC50 = 4800 nM T57392 CV31WQ 44449136 IC50 = 3200 nM T57392 CA4DS0 44449171 IC50 = 820 nM T57392 CA61WE 44449202 IC50 = 3700 nM T57392 CC19LO 44449228 IC50 = 2300 nM T57392 C3RMF8 44449236 IC50 > 10000 nM T57392 C80CWR 44452935 IC50 = 610 nM T57392 CPM4W2 44454303 IC50 = 5100 nM T57392 CL6KS1 44454834 IC50 > 5000 nM T57392 CZ39GO 44455035 IC50 > 10000 nM T57392 CC87TA 44455458 IC50 = 1500 nM T57392 C68MTP 44455459 IC50 = 1300 nM T57392 CN1U6E 44455460 IC50 = 500 nM T57392 C0V4OX 44455461 IC50 = 17000 nM T57392 CDK31X 44455482 IC50 = 900 nM T57392 CI0K4G 44455483 IC50 = 22000 nM T57392 C8WZB6 44455484 IC50 = 4600 nM T57392 CYFI71 44455485 IC50 = 1600 nM T57392 CZE05M 44455509 IC50 = 800 nM T57392 CMS92F 44455510 IC50 = 200 nM T57392 CN60DZ 44455511 IC50 = 1300 nM T57392 C6OPJ8 44455539 IC50 = 400 nM T57392 C7O0AS 44455560 IC50 = 500 nM T57392 C4GOE6 44455625 IC50 = 800 nM T57392 CW1B8D 44455658 IC50 = 3300 nM T57392 CX0B5K 44455683 IC50 = 5900 nM T57392 CTV5H2 44455686 IC50 = 4700 nM T57392 C2F6XP 44455711 IC50 = 2500 nM T57392 CHCU69 44455744 IC50 = 3500 nM T57392 CA6L8Y 44455745 IC50 = 3100 nM T57392 CH67DO 44455765 IC50 = 500 nM T57392 CVH5R0 44455766 IC50 = 2200 nM T57392 CD5U7E 44455767 IC50 = 16000 nM T57392 CMC9H4 44455788 IC50 = 1400 nM T57392 CM3R2V 44455790 IC50 = 400 nM T57392 CCD6Q4 44455791 IC50 = 3800 nM T57392 C71TBV 44455792 IC50 = 200 nM T57392 CYF74A 44455793 IC50 = 7000 nM T57392 C2BML0 44455817 IC50 = 4000 nM T57392 C53JVI 44455818 IC50 = 600 nM T57392 C7MH1U 44455819 IC50 > 100000 nM T57392 C8B0KA 44455820 IC50 = 1000 nM T57392 CP3KW7 44455841 IC50 = 300 nM T57392 CQ2KX1 44455844 IC50 = 500 nM T57392 C0A6GB 44455845 IC50 = 8200 nM T57392 C6T5ZS 44455846 IC50 = 3000 nM T57392 CIVE78 44455847 IC50 = 2800 nM T57392 CU6AX0 44455869 IC50 = 2100 nM T57392 CN0JV1 44455871 IC50 = 900 nM T57392 C28WVU 44455872 IC50 = 3500 nM T57392 CWL42H 44457199 IC50 = 24000 nM T57392 CL9O8M 44462783 IC50 = 2000 nM T57392 C2QK4J 44472590 IC50 = 2200 nM T57392 CQ8C3F 44472591 IC50 = 31000 nM T57392 CWN95E 44472610 IC50 > 100000 nM T57392 C1H2ZT 44472612 IC50 = 39000 nM T57392 CM37YN 44475195 IC50 > 10 nM T57392 CSBL94 44475353 IC50 > 10 nM T57392 C3GYC0 44475943 IC50 >= 100000 nM T57392 CX9TJ4 44476890 IC50 > 50000 nM T57392 CUA9F0 44512094 IC50 > 50000 nM T57392 C1ED8S 44512617 IC50 = 29000 nM T57392 C4M9FH 44512619 IC50 = 29000 nM T57392 CU80BP 44517743 IC50 > 21000 nM T57392 CS9H0L 44517795 IC50 > 50000 nM T57392 CKI82C 44518336 IC50 > 1000 nM T57392 CSO35V 44520546 IC50 > 10000 nM T57392 CJCB39 44520861 IC50 = 8900 nM T57392 CJA36X 44533150 IC50 = 13000 nM T57392 C9N1BU 44539192 IC50 > 20000 nM T57392 C14SNF 44539764 IC50 > 30000 nM T57392 CLMY52 44539967 IC50 = 6900 nM T57392 CMW56J 44539973 IC50 > 30000 nM T57392 C0RA9E 44540072 IC50 > 30000 nM T57392 CV92IJ 44541354 IC50 = 52 nM T57392 C27TZY 44543970 IC50 = 41000 nM T57392 CK1Z8P 44545482 IC50 > 50000 nM T57392 CECD12 44547033 IC50 = 1800 nM T57392 CX13MK 44547414 IC50 > 50000 nM T57392 CP6R2X 44551848 IC50 = 36000 nM T57392 C4RB7W 44555352 IC50 > 10000 nM T57392 C5EX1K 44555473 IC50 > 10000 nM T57392 CVJ8S4 44559524 IC50 > 100000 nM T57392 CCGE36 44559528 IC50 > 100000 nM T57392 C32AGV 44561123 IC50 = 160 nM T57392 CG1W8A 44561157 IC50 = 5900 nM T57392 CXH86I 44561195 IC50 = 16000 nM T57392 CD7A4H 44561196 IC50 = 33000 nM T57392 C8HCR6 44561197 IC50 = 33000 nM T57392 C9HG8L 44561236 IC50 = 33000 nM T57392 CR5T0L 44561237 IC50 = 33000 nM T57392 CF21JK 44561238 IC50 = 6200 nM T57392 CMJ60R 44561239 IC50 = 3500 nM T57392 C0W4HQ 44561240 IC50 = 30000 nM T57392 C6A0TH 44561276 IC50 = 17000 nM T57392 CP7RQ8 44562623 IC50 = 4000 nM T57392 CHE68Z 44562624 IC50 = 3300 nM T57392 CR4TG7 44562625 IC50 = 4000 nM T57392 CH32FI 44562626 IC50 = 2000 nM T57392 CX1P3L 44562627 IC50 = 500 nM T57392 C0S8ZG 44562682 IC50 = 1400 nM T57392 C2HKE0 44562772 IC50 > 10000 nM T57392 C50WKO 44562773 IC50 = 4000 nM T57392 C3JD7Y 44562774 IC50 = 6500 nM T57392 CS0LD7 44562775 IC50 = 1500 nM T57392 C7AC8Z 44562776 IC50 = 1500 nM T57392 CU6G4W 44562777 IC50 = 1000 nM T57392 CCA0H2 44562815 IC50 = 1000 nM T57392 CQ0I5R 44562816 IC50 > 10000 nM T57392 CC1IF3 44562817 IC50 > 10000 nM T57392 CR28PD 44563213 IC50 = 600 nM T57392 CU4PD5 44563214 IC50 = 2000 nM T57392 CGKL94 44563257 IC50 = 400 nM T57392 C8TYL3 44563258 IC50 = 900 nM T57392 C8XUD6 44563259 IC50 = 5000 nM T57392 CIG6Z4 44563260 IC50 = 1300 nM T57392 C9VFW6 44563261 IC50 > 10000 nM T57392 CV1IL5 44565796 IC50 > 10000 nM T57392 C8DUG3 44566070 EC50 > 100000 nM T57392 CJB91U 44568803 IC50 > 25000 nM T57392 CR7C6A 44568804 IC50 > 25000 nM T57392 CQ7SL3 44568819 IC50 > 25000 nM T57392 C1OVN0 44568820 IC50 > 25000 nM T57392 CB5S9R 44569927 IC50 = 28000 nM T57392 C6Q5DK 44569945 IC50 = 89000 nM T57392 CBET53 44570224 IC50 = 36000 nM T57392 CP32DL 44570256 IC50 = 42000 nM T57392 CVO8L1 44570275 IC50 = 20000 nM T57392 C1MDQ6 44570537 IC50 = 4300 nM T57392 CAP51K 44570583 IC50 = 33000 nM T57392 C1W9AF 44570584 IC50 = 17000 nM T57392 CI1ZL9 44570617 IC50 = 21000 nM T57392 CZ56HX 44574108 IC50 > 5000 nM T57392 CN5WP4 44574711 IC50 > 10000 nM T57392 C3NKY2 44577989 Ki = 70 nM T57392 CFJB16 44578266 IC50 = 3100 nM T57392 CE54ZK 44578267 IC50 = 1890 nM T57392 CSFE81 44578268 IC50 = 185 nM T57392 CQ30GC 44578271 IC50 = 350 nM T57392 C8HB0Z 44578272 IC50 = 5360 nM T57392 CH3U5D 44578314 IC50 = 350 nM T57392 C17YVO 44578319 IC50 = 840 nM T57392 C8AP4K 44578374 IC50 = 420 nM T57392 CG80OC 44578914 IC50 > 50000 nM T57392 C7LAT0 44578954 IC50 > 50000 nM T57392 CBG04P 44578955 IC50 > 50000 nM T57392 CA3FO8 44578956 IC50 = 4900 nM T57392 CA16QJ 44578957 IC50 > 50000 nM T57392 CFH01N 44578958 IC50 > 50000 nM T57392 CMA26F 44578959 IC50 > 50000 nM T57392 C79PYS 44578960 IC50 > 50000 nM T57392 CF39ON 44578961 IC50 > 50000 nM T57392 C4KI0B 44579189 IC50 > 50000 nM T57392 C1I0QG 44579190 IC50 > 50000 nM T57392 C6VFZ3 44579191 IC50 > 50000 nM T57392 C1O5ET 44579232 IC50 > 50000 nM T57392 CY8NJ4 44579233 IC50 > 50000 nM T57392 CSLC36 44579234 IC50 > 50000 nM T57392 CBK23W 44579235 IC50 > 50000 nM T57392 CS2KV6 44579236 IC50 > 50000 nM T57392 C60CAD 44579237 IC50 > 50000 nM T57392 CX85MD 44579273 IC50 > 50000 nM T57392 C3L5ER 44583033 IC50 = 1.26 nM T57392 C0IP7C 44583234 IC50 > 10000 nM T57392 C6HTC1 44583235 IC50 > 10000 nM T57392 CZJU04 44583236 IC50 > 10000 nM T57392 C3TYW0 44583237 IC50 > 10000 nM T57392 CCL9R0 44583238 IC50 > 10000 nM T57392 COX7F1 44583287 IC50 < 10000 nM T57392 C5SI9Q 44583288 IC50 > 10000 nM T57392 CFT74N 44583289 IC50 > 10000 nM T57392 CC19TZ 44583290 IC50 > 10000 nM T57392 C90RAV 44583349 IC50 > 10000 nM T57392 CK81NJ 44583350 IC50 > 10000 nM T57392 C20VTN 44583351 IC50 > 10000 nM T57392 CD5U3A 44583352 IC50 > 10000 nM T57392 C9G7VT 44583353 IC50 > 10000 nM T57392 C6QF4O 44583354 IC50 > 10000 nM T57392 C48AQR 44583355 IC50 = 10000 nM T57392 CG5X0M 44583356 IC50 < 10000 nM T57392 CUG9Y0 44583357 IC50 > 10000 nM T57392 CRE9Q2 44583561 IC50 = 41000 nM T57392 C9AP1O 44583590 IC50 > 100000 nM T57392 C5IUL8 44587443 IC50 = 4100 nM T57392 C59KDV 44587445 IC50 = 440 nM T57392 CLCE75 44587446 IC50 = 12000 nM T57392 CPF01B 44587447 IC50 = 5800 nM T57392 CIL89C 44587448 IC50 = 5700 nM T57392 CF0I6D 44587449 IC50 = 1400 nM T57392 C0J4LS 44587450 IC50 = 880 nM T57392 CY0F1M 44587482 IC50 = 1400 nM T57392 CL5M2J 44587483 IC50 = 180 nM T57392 CRN0Z1 44587484 IC50 = 5000 nM T57392 CTN0Q1 44587485 IC50 = 400 nM T57392 CAHW83 44587486 IC50 = 90 nM T57392 CJY60H 44587487 IC50 = 200 nM T57392 C3OL1M 44587488 IC50 = 70 nM T57392 C56QTZ 44587489 IC50 = 9000 nM T57392 CCS62T 44587583 IC50 = 199.53 nM T57392 C4WB1N 44589201 IC50 = 1800 nM T57392 C9RA0C 44589548 EC50 > 50000 nM T57392 CH54CO 44589824 IC50 = 9120 nM T57392 C89LHN 44589825 IC50 = 2730 nM T57392 CPH6S0 44593451 IC50 = 800 nM T57392 C3ZI2Y 44593546 IC50 = 40000 nM T57392 C6PEV1 44593547 IC50 = 5900 nM T57392 C70MSI 44593549 IC50 = 96000 nM T57392 C0IE3Y 44593553 IC50 = 2100 nM T57392 C9F6EB 44593557 IC50 = 6600 nM T57392 CAWE52 44593632 Ki = 660 nM T57392 CP37YX 44593633 Ki = 20 nM T57392 C29QEV 44593636 Ki = 120 nM T57392 CCA7K5 44593648 IC50 > 50000 nM T57392 C64ZKC 44593664 IC50 > 10000 nM T57392 C01BFQ 44593665 IC50 > 10000 nM T57392 C1DI5Z 44593686 IC50 = 1200 nM T57392 C7YLS4 44593687 IC50 = 1600 nM T57392 C6KGF2 44593688 IC50 = 800 nM T57392 CU8F9L 44593689 IC50 = 210 nM T57392 CR18ZA 44593690 IC50 = 370 nM T57392 C20YZD 44593691 IC50 = 4000 nM T57392 CN52LH 44593692 IC50 = 700 nM T57392 C7IU8S 44593694 IC50 = 800 nM T57392 C9SM4D 44593695 IC50 = 800 nM T57392 CSQ14O 44593696 IC50 = 310 nM T57392 CE97GB 44596160 IC50 > 20000 nM T57392 C4ID9A 44602971 IC50 = 300 nM T57392 C7I4EY 44603096 IC50 > 30000 nM T57392 C4MOE2 44603271 IC50 > 10000 nM T57392 C89VRG 44605616 IC50 > 10000 nM T57392 CZD25I 44605617 IC50 > 10000 nM T57392 CXQ19C 44610104 IC50 = 17000 nM T57392 C0WVZ1 44622338 IC50 > 30000 nM T57392 CL26YD 44622339 IC50 > 30000 nM T57392 CA7EQ2 44622340 IC50 > 30000 nM T57392 C23ORN 44622341 IC50 > 30000 nM T57392 C2JIX6 44622342 IC50 > 30000 nM T57392 CNI29G 44622416 IC50 > 30000 nM T57392 C9KUD5 44622417 IC50 > 30000 nM T57392 C4Q7JB 44622418 IC50 > 30000 nM T57392 C12SGH 44622499 IC50 > 30000 nM T57392 C2OUJ0 44624151 IC50 > 5000 nM T57392 COM81X 44625569 IC50 = 1995.26 nM T57392 C2D0TJ 44625571 IC50 = 3981.07 nM T57392 C0N6DO 44625908 IC50 > 50000 nM T57392 CXD90A 44625911 IC50 > 50000 nM T57392 C85ZIF 44626928 IC50 > 10000 nM T57392 C4BYG5 44626929 IC50 > 10000 nM T57392 CQE59L 44627133 IC50 > 10000 nM T57392 CDQ47G 44629236 IC50 > 25000 nM T57392 CH3SF9 44631836 IC50 > 27000 nM T57392 CPG61Y 44718445 IC50 = 13000 nM T57392 C3Q7BW 44816514 IC50 > 30000 nM T57392 C85DWU 44816692 IC50 > 30000 nM T57392 CJ0F5Q 44819015 IC50 > 30000 nM T57392 CN21OS 44819193 IC50 > 30000 nM T57392 C65KPR 45101722 IC50 = 19600 nM T57392 CQI0D4 45102707 IC50 = 200 nM T57392 CSEP-69 45102708 IC50 < 1000 nM T57392 CGCZ64 45102767 IC50 > 50000 nM T57392 C7NFZ1 45110765 IC50 > 30000 nM T57392 CUL67Y 45202552 IC50 = 27100 nM T57392 C4IY8M 45256689 IC50 > 50000 nM T57392 C1K0ZH 45259193 IC50 = 3981.07 nM T57392 CB9QZ6 45263405 IC50 = 500 nM T57392 CQ85WF 45263621 IC50 = 1100 nM T57392 CUT2B4 45267348 IC50 > 10000 nM T57392 C8H9GV 45267527 IC50 = 700 nM T57392 CP9B0W 45267530 IC50 = 5000 nM T57392 C3GJK0 45267531 IC50 = 2200 nM T57392 C6SV5O 45267774 Ki = 1036 nM T57392 CHQ05B 45267775 IC50 > 20000 nM T57392 C53DIE 45267853 IC50 > 30000 nM T57392 CJH3A2 45268206 IC50 > 10000 nM T57392 C0QB1V 45268417 IC50 = 1800 nM T57392 C2S9ZT 45268436 IC50 = 14200 nM T57392 CULJ91 45268456 IC50 > 30000 nM T57392 CSJ4L2 45268478 IC50 > 3000 nM T57392 C9B5EH 45268653 IC50 = 35150 nM T57392 C65LBY 45268662 Ki = 502 nM T57392 CUQ23Z 45268922 IC50 = 600 nM T57392 C4WR0V 45269087 IC50 > 10000 nM T57392 CRPS25 45269096 IC50 > 10000 nM T57392 C7BNY6 45269104 IC50 > 10000 nM T57392 C9HR0K 45269274 IC50 = 100 nM T57392 CZ1N2O 45269275 IC50 = 12400 nM T57392 CIE21V 45269276 IC50 > 25000 nM T57392 CB5O6V 45269307 IC50 > 30000 nM T57392 CF2P9H 45269325 IC50 > 30000 nM T57392 CCFG82 45269436 IC50 = 6360 nM T57392 CS1Q2X 45269947 IC50 > 10000 nM T57392 C1BE5U 45269948 IC50 > 10000 nM T57392 CG1H9N 45269950 IC50 > 10000 nM T57392 C8QJ7X 45270108 IC50 = 100 nM T57392 CYWK62 45270115 IC50 = 1700 nM T57392 C03ETI 45270148 IC50 > 30000 nM T57392 C3GA6N 45270158 IC50 = 3170 nM T57392 C6YI5N 45270172 IC50 > 30000 nM T57392 C57TQW 45270199 IC50 = 29000 nM T57392 C8GQ7J 45270330 IC50 = 16309 nM T57392 C48BMQ 45270339 IC50 = 4353 nM T57392 CFZ01K 45270350 IC50 = 360 nM T57392 COFD89 45270589 IC50 = 2400 nM T57392 C1NT2M 45270771 IC50 > 10000 nM T57392 CA05IG 45270778 IC50 > 10000 nM T57392 CZ7MK9 45270788 IC50 > 10000 nM T57392 CGF7Z6 45270958 IC50 = 3600 nM T57392 CH5S8Y 45270959 IC50 > 25000 nM T57392 CY70SI 45270983 IC50 > 30000 nM T57392 C2XH3A 45270987 IC50 > 30000 nM T57392 CU9HV3 45271001 IC50 = 430 nM T57392 C18WQE 45271166 IC50 = 7319 nM T57392 CW6HL5 45271167 Ki = 805 nM T57392 C9TM2P 45271593 IC50 > 10000 nM T57392 C06YAD 45271599 IC50 > 10000 nM T57392 CG0I8P 45271610 IC50 > 10000 nM T57392 C6FBH0 45271618 IC50 > 10000 nM T57392 C5NH6Q 45271791 IC50 = 900 nM T57392 C8Z3DK 45271794 IC50 = 400 nM T57392 CX62YA 45271796 IC50 > 25000 nM T57392 CZ8EO2 45271803 IC50 > 25000 nM T57392 CJ7Q9E 45271813 IC50 = 6300 nM T57392 CU9C4I 45272046 IC50 = 4444 nM T57392 CAY8I7 45272070 IC50 = 1480 nM T57392 C71VIG 45272510 IC50 > 10000 nM T57392 C05EDY 45272511 IC50 > 10000 nM T57392 CJI2R6 45272664 IC50 = 4300 nM T57392 C49BKQ 45272672 IC50 = 3900 nM T57392 CP36CT 45272682 IC50 = 1300 nM T57392 C8NL4U 45272683 IC50 = 100 nM T57392 C35DUQ 45272700 IC50 > 30000 nM T57392 CKUI32 45272704 IC50 > 30000 nM T57392 C62IGT 45272875 IC50 = 12798 nM T57392 C3GUK4 45272876 IC50 = 7210 nM T57392 CBE0M8 45272877 IC50 = 6072 nM T57392 CR04WH 45272878 IC50 = 8185 nM T57392 CZ7N8Q 45272889 IC50 = 12134 nM T57392 CK2B5U 45272890 IC50 = 6134 nM T57392 C8TC4R 45272894 IC50 = 1117 nM T57392 CA0SD1 45272895 IC50 = 5219 nM T57392 CUK91L 45273154 IC50 = 5500 nM T57392 CD62AH 45273373 IC50 > 10000 nM T57392 CMN39U 45273380 IC50 > 10000 nM T57392 CYMR87 45273573 IC50 = 4600 nM T57392 CFL87A 45273581 IC50 = 800 nM T57392 C2XB0P 45273589 IC50 = 1700 nM T57392 C28PRV 45273594 IC50 > 25000 nM T57392 CSX2T9 45273602 IC50 = 11600 nM T57392 CMP59Q 45273603 IC50 = 1100 nM T57392 C3U7KT 45273637 IC50 > 30000 nM T57392 C5E2XR 45273828 IC50 = 1534 nM T57392 CE71LQ 45273833 Ki = 2053 nM T57392 CZ71RN 45278805 IC50 > 20000 nM T57392 CYOW10 45377016 IC50 > 50000 nM T57392 C7D3LB 45377018 IC50 = 20325 nM T57392 C25PTU 45377580 IC50 = 3775 nM T57392 C8ELI4 45378010 IC50 = 392 nM T57392 CMU6Z8 45379828 IC50 > 6000 nM T57392 CNQT48 45379947 IC50 = 1000 nM T57392 CLK8O9 45380748 IC50 = 6000 nM T57392 C84ORB 45380848 IC50 > 20000 nM T57392 C0CHF4 45482789 IC50 > 10000 nM T57392 CZUI01 45484860 IC50 > 5000 nM T57392 C65ONH 45484861 IC50 > 5000 nM T57392 C6KC8V 45484873 IC50 > 5000 nM T57392 CVR40A 45484874 IC50 > 5000 nM T57392 CV78NM 45484881 IC50 > 5000 nM T57392 C5DEA7 45484892 IC50 > 5000 nM T57392 CXYK82 45484893 IC50 > 5000 nM T57392 CR8VF3 45484894 IC50 > 5000 nM T57392 C7TQ3Z 45484899 IC50 > 5000 nM T57392 CD7N4J 45484900 IC50 > 5000 nM T57392 CQ84RV 45484907 IC50 > 5000 nM T57392 C1K0IO 45484913 IC50 > 5000 nM T57392 C2J4VM 45484915 IC50 > 5000 nM T57392 CE6J7S 45484916 IC50 > 5000 nM T57392 CI4SP9 45484917 IC50 > 5000 nM T57392 CYA6U2 45484918 IC50 > 5000 nM T57392 CYWT18 45484919 IC50 > 5000 nM T57392 C1FZ3N 45484922 IC50 > 5000 nM T57392 CXD74W 45484923 IC50 > 5000 nM T57392 CDP3X6 45484930 IC50 > 5000 nM T57392 CQ90DC 45484931 IC50 > 5000 nM T57392 CQ3I9D 45484949 IC50 > 5000 nM T57392 CZU29D 45484950 IC50 > 5000 nM T57392 CW6M7Q 45484961 IC50 > 5000 nM T57392 C4TI0X 45484966 IC50 > 5000 nM T57392 CWNH93 45484967 IC50 > 5000 nM T57392 C5R0YZ 45484968 IC50 > 5000 nM T57392 C9E4UO 45484969 IC50 > 5000 nM T57392 CL32NJ 45488686 IC50 > 10000 nM T57392 C7UAT9 46174270 IC50 > 30000 nM T57392 CB0J1G 46174396 IC50 = 900 nM T57392 CPU02J 46190696 IC50 = 7367 nM T57392 CQDI48 46191427 IC50 > 20000 nM T57392 CAT9Z8 46191428 IC50 > 20000 nM T57392 CP08ZD 46191499 IC50 > 20000 nM T57392 C0ET7O 46191501 IC50 = 19000 nM T57392 C4HSX5 46191502 IC50 = 17000 nM T57392 CSD13A 46191565 IC50 = 11000 nM T57392 CXIC58 46191567 IC50 = 4900 nM T57392 C71CGU 46191622 IC50 < 80 nM T57392 CFYP54 46203897 IC50 = 1400 nM T57392 C21ICG 46212134 IC50 > 50000 nM T57392 CN3BE0 46212588 IC50 > 20000 nM T57392 CC9X1M 46213938 IC50 = 13200 nM T57392 CPF0J9 46214673 IC50 > 30000 nM T57392 CAX31B 46216689 IC50 > 15000 nM T57392 CL51NF 46216732 IC50 = 7100 nM T57392 CZJL95 46216733 IC50 > 10000 nM T57392 C5AY6M 46220498 IC50 > 10000 nM T57392 CFS6Q5 46224644 IC50 = 15000 nM T57392 CURS28 46224649 IC50 = 25000 nM T57392 C75QAG 46224653 IC50 = 9000 nM T57392 CB5HP0 46224657 IC50 = 13000 nM T57392 CI3OC4 46224664 IC50 = 13000 nM T57392 CS9D6X 46224668 IC50 = 7300 nM T57392 C5N2WP 46224669 IC50 = 20000 nM T57392 C6XQF5 46224670 IC50 = 10000 nM T57392 C72ZGS 46224672 IC50 = 14000 nM T57392 CNG16S 46224673 IC50 > 33000 nM T57392 CS0Y7O 46224677 IC50 = 22000 nM T57392 CJP6A9 46224678 IC50 = 16000 nM T57392 CR9J1L 46224680 IC50 = 22000 nM T57392 CZS7L4 46224681 IC50 = 31000 nM T57392 CJZL72 46224683 IC50 > 33000 nM T57392 CKQF01 46224685 IC50 = 15000 nM T57392 C15RNW 46224687 IC50 = 6000 nM T57392 C81YIZ 46224688 IC50 = 13000 nM T57392 CRSM47 46224691 IC50 = 7500 nM T57392 C0RJG8 46224692 IC50 = 11000 nM T57392 CQC6J0 46224693 IC50 = 16000 nM T57392 C2A5QX 46224699 IC50 = 28000 nM T57392 CPHQ30 46224702 IC50 = 17000 nM T57392 C7JXG3 46224705 IC50 = 8000 nM T57392 CMYU19 46224706 IC50 = 7500 nM T57392 C1DO4U 46230960 IC50 > 10000 nM T57392 C59XOB 46230961 IC50 > 10000 nM T57392 C9EGU1 46230962 IC50 > 10000 nM T57392 C7G3TB 46231012 IC50 > 10000 nM T57392 C1J0WY 46231013 IC50 > 10000 nM T57392 CALC10 46231014 IC50 > 10000 nM T57392 C2FVA8 46231075 IC50 = 1800 nM T57392 CA3R5W 46231076 IC50 > 10000 nM T57392 CSZ2F6 46231077 IC50 = 1100 nM T57392 CVL6C0 46231146 IC50 = 1300 nM T57392 C8W4VL 46231147 IC50 = 100 nM T57392 CRTO63 46231148 IC50 = 1700 nM T57392 CZ6C0S 46231149 IC50 = 1100 nM T57392 C80DAS 46231312 IC50 < 10000 nM T57392 CVJU38 46233842 IC50 = 3700 nM T57392 CQ9A7L 46234188 IC50 > 30000 nM T57392 C94GCA 46234349 IC50 > 30000 nM T57392 C8PZU1 46235580 IC50 > 50 nM T57392 C7OB2G 46235733 IC50 = 2470 nM T57392 CIGB53 46237137 IC50 > 12 ug.mL-1 T57392 CQX93F 46398805 IC50 > 10000 nM T57392 CJ2D3O 46701015 IC50 = 6960 nM T57392 CM04ZI 46701016 IC50 = 4350 nM T57392 C0JWP5 46701017 IC50 = 5210 nM T57392 C5H0MJ 46701086 IC50 = 2650 nM T57392 C9HWI7 46701087 IC50 = 7930 nM T57392 CVE5O1 46701088 IC50 = 8000 nM T57392 C1VPM0 46701089 IC50 = 1100 nM T57392 CQ8B6R 46701090 IC50 = 2920 nM T57392 C6C0FS 46701091 IC50 = 250 nM T57392 CC68WI 46830289 IC50 > 10000000 nM T57392 C5TC2S 46830335 IC50 > 10000 nM T57392 C1K7FL 46830336 IC50 > 10000 nM T57392 C2M9XO 46835914 IC50 > 40000 nM T57392 C9CR0E 46835922 IC50 > 40000 nM T57392 C1N4KX 46842383 IC50 > 10000 nM T57392 CPE23Q 46850145 IC50 > 20000 nM T57392 C2UYK7 46850264 IC50 = 16000 nM T57392 CD04SA 46852212 IC50 > 3000 nM T57392 CT6MJ2 46852951 IC50 > 50000 nM T57392 CBZE98 46853681 IC50 > 30000 nM T57392 CO31WX 46861576 IC50 = 3600 nM T57392 CW1FS9 46861860 IC50 = 2500 nM T57392 C0EG8P 46865563 IC50 > 50000 nM T57392 C2QH7O 46865650 IC50 = 17000 nM T57392 CQN2H4 46865774 IC50 = 2700 nM T57392 CC5KR7 46865978 IC50 = 5600 nM T57392 C9T0ZE 46866390 IC50 > 30000 nM T57392 CO3P0J 46866604 IC50 > 30000 nM T57392 C8OY4U 46869951 IC50 > 30000 nM T57392 CCWK45 46871629 IC50 = 500 nM T57392 CLVI62 46879428 IC50 = 300 nM T57392 CL2A4H 46879430 IC50 < 100 nM T57392 C9VRO6 46879432 IC50 < 100 nM T57392 CFH9W8 46879490 IC50 < 100 nM T57392 CG68BI 46879549 IC50 > 33000 nM T57392 C9H1PK 46879550 IC50 = 600 nM T57392 CB02YQ 46879551 IC50 = 1900 nM T57392 CCM7T2 46879552 IC50 = 25000 nM T57392 C7EHZ9 46879553 IC50 = 60000 nM T57392 CVI5O7 46879596 IC50 = 700 nM T57392 CL05QN 46879597 IC50 = 18000 nM T57392 CYK18D 46879598 IC50 = 45500 nM T57392 CG9N6P 46879643 IC50 = 26000 nM T57392 CCK8A9 46880206 IC50 < 100 nM T57392 C2MC4K 46881463 IC50 = 1000 nM T57392 CSQ4C9 46881468 IC50 > 10000 nM T57392 C4BH9E 46882458 IC50 < 100 nM T57392 CJ50FM 46882459 IC50 = 16000 nM T57392 CERN34 46882461 IC50 = 7900 nM T57392 CQN87I 46882521 IC50 < 100 nM T57392 C56ULO 46882522 IC50 = 1300 nM T57392 CRZ95W 46882582 IC50 = 500 nM T57392 CHS14B 46882671 IC50 = 16000 nM T57392 CC05XO 46882712 IC50 < 100 nM T57392 CL3EI9 46882713 IC50 = 200 nM T57392 CZ15LN 46882714 IC50 = 100 nM T57392 CD24US 46882752 IC50 < 100 nM T57392 CAN69D 46882753 IC50 = 600 nM T57392 CBXT24 46882756 IC50 = 1700 nM T57392 C39WEJ 46882794 IC50 = 1600 nM T57392 C4OZ1U 46882796 IC50 = 1100 nM T57392 CDK0Q3 46882797 IC50 = 300 nM T57392 CRU1P2 46882874 IC50 = 10000 nM T57392 CYU8X6 46882875 IC50 > 10000 nM T57392 CX5CZ7 46882876 IC50 < 10000 nM T57392 CC1VO9 46882918 IC50 > 10000 nM T57392 C27RIV 46882919 IC50 > 10000 nM T57392 CE3O7D 46882949 IC50 = 10000 nM T57392 CHS1X0 46882950 IC50 > 10000 nM T57392 C3S9WE 46882951 IC50 > 10000 nM T57392 C3A1ZF 46882969 IC50 < 10000 nM T57392 CG3D0K 46882971 IC50 > 10000 nM T57392 CD7XA2 46882972 IC50 > 10000 nM T57392 CY5CW2 46882973 IC50 > 10000 nM T57392 C3ZPY7 46882986 IC50 > 10000 nM T57392 CKX8N2 46882987 IC50 > 10000 nM T57392 CG81CZ 46882988 IC50 > 10000 nM T57392 CP87CA 46883032 IC50 > 10000 nM T57392 CWU4T2 46883033 IC50 > 10000 nM T57392 C41RYD 46883034 IC50 > 10000 nM T57392 C3SQ2Z 46883035 IC50 > 10000 nM T57392 CS51UC 46883473 IC50 > 10000 nM T57392 CL0S4B 46883474 IC50 > 10000 nM T57392 C0K5ZJ 46883508 IC50 > 10000 nM T57392 CMNJ24 46883509 IC50 > 10000 nM T57392 CF4VC1 46883510 IC50 = 10000 nM T57392 CW6A9I 46884062 IC50 = 9.8 nM T57392 C04JMO 46884063 IC50 > 10000 nM T57392 CR0CQ9 46884120 IC50 = 9500 nM T57392 C9OYT5 46884152 IC50 = 4000 nM T57392 CCI32B 46884153 IC50 = 1500 nM T57392 C20HET 46884155 IC50 > 10000 nM T57392 C0HYN3 46884200 IC50 = 9500 nM T57392 CM6A8S 46884201 IC50 = 4926000 nM T57392 CW94IK 46884202 IC50 > 10000000 nM T57392 C3QT0U 46884239 IC50 = 8012000 nM T57392 COPQ16 46884600 IC50 = 6000 nM T57392 C85MOA 46884637 IC50 = 22000 nM T57392 C36NKV 46884638 IC50 = 3200 nM T57392 CQ84IF 46884639 IC50 = 900 nM T57392 CZGS15 46884640 IC50 > 10000 nM T57392 CZ72SW 46884641 IC50 > 10000 nM T57392 CA3Z6G 46884666 IC50 = 3800 nM T57392 C8DBY0 46884667 IC50 > 10000 nM T57392 CU3BG6 46884668 IC50 = 6600 nM T57392 CPG14Q 46884669 IC50 = 5300 nM T57392 C7R9AK 46884670 IC50 = 36000 nM T57392 C64KNW 46884698 IC50 = 690 nM T57392 C0ASK4 46884699 IC50 = 22000 nM T57392 CYNU85 46884731 IC50 = 12000 nM T57392 CJ6O8D 46884732 IC50 = 11000 nM T57392 C9QT7G 46884733 IC50 = 1900 nM T57392 CL6Z7Q 46884734 IC50 = 6400 nM T57392 C6PRX8 46884735 IC50 = 1000 nM T57392 CWK8I4 46884736 IC50 = 1400 nM T57392 CB8GE1 46884818 IC50 > 10000 nM T57392 C4MQ0A 46884856 IC50 > 10000 nM T57392 CCNT25 46884898 IC50 > 10000 nM T57392 C3MSG2 46885027 IC50 > 10000 nM T57392 CB7XI0 46885213 IC50 > 10000 nM T57392 CRE96X 46885625 IC50 < 100 nM T57392 CM76UZ 46888550 IC50 > 12 ug.mL-1 T57392 CJK1Z5 46888857 IC50 = 2300 nM T57392 CX92WH 46889257 IC50 > 10000 nM T57392 C01DMO 46889258 IC50 > 10000 nM T57392 CX18GT 46889932 IC50 > 10000 nM T57392 CI14SE 46890441 IC50 > 30000 nM T57392 CZ2MG7 46890444 IC50 = 17700 nM T57392 CD5J8B 46890446 IC50 = 12100 nM T57392 CZ90FC 46894119 IC50 > 30000 nM T57392 CC4GA0 46895367 IC50 = 25000 nM T57392 C90NYX 46896338 IC50 = 5000 nM T57392 CC9FZ0 46898063 IC50 > 20 nM T57392 C1JSH9 46899637 IC50 > 10000 nM T57392 CV3LP2 46899639 IC50 > 6000 nM T57392 CGHZ15 46899640 IC50 > 10000 nM T57392 CWR9M5 46900138 IC50 > 10000 nM T57392 CGN7Q8 46900139 IC50 > 10000 nM T57392 CP41AQ 46900457 IC50 < 1000 nM T57392 CR3L4I 46900459 IC50 > 10000 nM T57392 CK17PA 46900606 IC50 > 5000 nM T57392 C1NAX4 46900612 IC50 > 5000 nM T57392 CXD9S3 46900776 IC50 > 10000 nM T57392 C7QDM9 46900782 IC50 > 8000 nM T57392 C15FMY 46900954 IC50 > 7000 nM T57392 C3JCB1 46911060 IC50 > 50000 nM T57392 CHUV97 46911229 IC50 > 5000 nM T57392 CXJ7M5 46911719 IC50 = 41750 nM T57392 CA2GO4 46911720 IC50 > 45000 nM T57392 C1VA0B 46912953 IC50 > 5000 nM T57392 CN9L7G 46916268 IC50 > 10000 nM T57392 CLV1W2 46918487 IC50 > 10000 nM T57392 C65QAB 46927297 IC50 > 10000 nM T57392 C47HDL 46929447 IC50 = 9500 nM T57392 CSDO60 46929548 IC50 = 3600 nM T57392 C6F2MP 46929551 IC50 = 820 nM T57392 CZJ2G8 46929554 IC50 = 4300 nM T57392 CKO76R 46931815 IC50 > 5000 nM T57392 C68AJP 46933238 IC50 = 600 nM T57392 CV98OS 46933385 IC50 = 10500 nM T57392 C0J8WS 46933530 IC50 > 20000 nM T57392 CJK53D 46933697 IC50 > 100000 nM T57392 CAY75I 46934585 IC50 = 10000 nM T57392 CU90MG 46938037 IC50 > 20000000 nM T57392 CX2U5I 46938097 IC50 > 20000000 nM T57392 C47QBL 46938101 IC50 > 20000000 nM T57392 C9DLV2 46945057 IC50 > 50000 nM T57392 CZ0G6A 46947062 IC50 = 17380 nM T57392 CF14PE 46947264 IC50 > 30000 nM T57392 CX6NK2 47144386 IC50 = 50000 nM T57392 CBV0H3 49765039 IC50 > 10000 nM T57392 CWU2R3 49773361 IC50 > 40000 nM T57392 C9RI3L 49780809 IC50 > 4000 nM T57392 CYL65E 49781476 IC50 > 10000 nM T57392 CY1OJ5 49797177 IC50 > 30000 nM T57392 CON0A6 49797232 IC50 = 950 nM T57392 CA4E8M 49797242 IC50 = 11600 nM T57392 C37MDP 49797244 IC50 = 100 nM T57392 CUMH43 49797248 IC50 = 16200 nM T57392 C6DJX7 49797605 IC50 = 1500 nM T57392 C85KNS 49798241 IC50 = 1050 nM T57392 CQ4G1V 49798242 IC50 = 4000 nM T57392 C01JNE 49798243 IC50 = 8260 nM T57392 CC6MF8 49798244 IC50 = 9100 nM T57392 CYAS45 49798266 IC50 = 4700 nM T57392 CQVG17 49798349 IC50 = 53703.18 nM T57392 C62VRQ 49798437 IC50 > 100000 nM T57392 CY90CD 49798461 IC50 > 100000 nM T57392 CF8J6E 49798462 IC50 > 100000 nM T57392 C02EUQ 49800098 IC50 > 10000 nM T57392 C9YSF2 49800475 IC50 > 30000 nM T57392 CD8KX3 49804491 IC50 > 30000 nM T57392 CET89N 49822116 IC50 > 20000 nM T57392 CVS85M 49831162 IC50 > 10000 nM T57392 COM5Q7 49836030 IC50 > 40000 nM T57392 CT7CV0 49836295 IC50 > 10000 nM T57392 CYJW87 49836299 IC50 > 10000 nM T57392 C8E6WA 49836410 IC50 > 10000 nM T57392 CNM9X8 49836528 IC50 > 10000 nM T57392 COK75S 49836633 IC50 > 10000 nM T57392 CB81YG 49836637 IC50 > 10000 nM T57392 CD8GN9 49837170 EC50 > 100000 nM T57392 CB71TA 49837867 IC50 > 50000 nM T57392 CZQC64 49837869 IC50 = 50000 nM T57392 CVNA15 49837870 IC50 = 50000 nM T57392 C9L3XR 49838879 IC50 > 13000 nM T57392 C06MKW 49839561 IC50 > 10000 nM T57392 C3DN7U 49843520 IC50 > 10000 nM T57392 CECB91 49843530 IC50 > 31000 nM T57392 CF91RS 49843531 IC50 = 9510 nM T57392 CY46CB 49843532 IC50 > 50000 nM T57392 CU63QR 49847377 IC50 > 50000 nM T57392 CZT4I8 49847378 IC50 > 50000 nM T57392 CA72PE 49847379 IC50 > 50000 nM T57392 C8KQB9 49848139 IC50 > 10000 nM T57392 C4V7EW 49848258 IC50 > 10000 nM T57392 C4BXP1 49848557 IC50 > 50000 nM T57392 CQ32CR 49848656 IC50 > 10000 nM T57392 CP8TS6 49848895 IC50 > 50000 nM T57392 C9COF5 49848896 IC50 > 50000 nM T57392 CK0B1G 49848897 IC50 > 50000 nM T57392 CP61VJ 49849002 IC50 > 50000 nM T57392 CBM62Z 49849007 IC50 > 50000 nM T57392 C05SEW 49849008 IC50 > 50000 nM T57392 CF64IJ 49849120 IC50 > 50000 nM T57392 CC9EB4 49849122 IC50 > 50000 nM T57392 C2ORV5 49849123 IC50 > 50000 nM T57392 CTR7Q0 49850345 IC50 > 50118.72 nM T57392 C8LBU5 49855513 IC50 > 30000 nM T57392 C5LY6T 49855593 IC50 = 10000 nM T57392 CQ0L4M 49856084 IC50 > 30000 nM T57392 C9TO2S 49856484 IC50 > 8900 nM T57392 C0N7RV 49856926 IC50 > 50000 nM T57392 C6POK9 49856931 IC50 = 10000 nM T57392 CC8VZ4 49857811 IC50 > 30000 nM T57392 CZO5D6 49857998 IC50 > 30000 nM T57392 CL93VT 49860116 Ki = 25000 nM T57392 C6O4ZK 49862647 IC50 > 5000 nM T57392 CGYM04 49864794 IC50 > 20000 nM T57392 C1I5PF 49864901 IC50 > 20000 nM T57392 CA4H2I 49864902 IC50 = 1900 nM T57392 CNFL69 49864903 IC50 > 20000 nM T57392 CY7U2X 49864936 IC50 > 20000 nM T57392 C8P2HI 49864937 IC50 > 20000 nM T57392 C8X3SL 49864938 IC50 > 20000 nM T57392 C2RN6C 49864988 IC50 = 20000 nM T57392 C59QLI 49864989 IC50 > 20000 nM T57392 CD29IW 49865043 IC50 = 1600 nM T57392 C6XT5M 49865104 IC50 = 9100 nM T57392 CBMQ90 49865105 IC50 = 6700 nM T57392 CMS6R4 49865106 IC50 = 4200 nM T57392 C0Y5ZU 49865137 IC50 > 20 nM T57392 C6GJ0L 49865162 IC50 = 5800 nM T57392 CA0RS7 49865163 IC50 = 5600 nM T57392 C3WTC1 49865164 IC50 = 20000 nM T57392 CG98LM 49865191 IC50 > 20 nM T57392 CR4F9G 49865290 IC50 = 1400 nM T57392 CFZ39O 49865822 IC50 = 2000 nM T57392 CT34HY 49865823 IC50 = 12000 nM T57392 CK7O1S 49865875 IC50 = 7000 nM T57392 CCH8T4 49865876 IC50 = 12000 nM T57392 C8V3NG 49865877 IC50 = 14000 nM T57392 CEK89Q 49865878 IC50 = 15000 nM T57392 CZA5X4 49865879 IC50 = 6000 nM T57392 CD4LO5 49865880 IC50 = 8000 nM T57392 C3YJ4G 49865936 IC50 = 300 nM T57392 CB5WR8 49865937 IC50 = 30 nM T57392 C0S8XD 49865953 IC50 = 33000 nM T57392 C8LJ4H 49865983 IC50 = 12000 nM T57392 C1MPT6 49865984 IC50 = 23000 nM T57392 C62NWE 49865985 IC50 = 600 nM T57392 C5H4AY 49865986 IC50 = 9000 nM T57392 C90XRC 49865987 IC50 = 15000 nM T57392 CEFJ14 49866038 IC50 = 3000 nM T57392 CZ9I3O 49866039 IC50 = 4000 nM T57392 C96XFK 49866040 IC50 = 36000 nM T57392 C26NLJ 49866041 IC50 = 14000 nM T57392 CQHM34 49866042 IC50 = 50 nM T57392 C8JY3K 49866095 IC50 = 13000 nM T57392 C9N5CZ 49866096 IC50 = 13000 nM T57392 CC1L4U 49866097 IC50 = 800 nM T57392 CV49QI 49866161 IC50 = 1000 nM T57392 CF59UG 49866162 IC50 = 4100 nM T57392 C5N8KG 49866163 IC50 = 40 nM T57392 C4F8UX 49866191 IC50 = 80 nM T57392 CMV6Y2 49868651 IC50 > 40000 nM T57392 C5OY7B 49872246 IC50 > 27000 nM T57392 C7GR0H 49872381 IC50 > 10000 nM T57392 CD1X3U 49872384 IC50 > 10000 nM T57392 C60RMP 49872483 IC50 = 16000 nM T57392 CV5BF3 49872645 IC50 > 27000 nM T57392 CN97FO 49872646 IC50 > 27000 nM T57392 CO0Y6K 49872677 IC50 > 10000 nM T57392 CD6P5R 49872735 IC50 > 27000 nM T57392 CL64NB 49872737 IC50 > 27000 nM T57392 CJWE29 49872771 IC50 > 10000 nM T57392 CK9VE4 49872772 IC50 > 10000 nM T57392 CFP14Q 49872867 IC50 > 10000 nM T57392 C83CTW 49872868 IC50 > 10000 nM T57392 CLB34U 49872872 IC50 > 10000 nM T57392 CAM1D0 49873181 IC50 > 10000 nM T57392 CFT6V9 49873225 IC50 = 600 nM T57392 CV1L4P 49873242 IC50 = 27000 nM T57392 C5BA2V 49873243 IC50 > 27000 nM T57392 CSN45W 49873329 IC50 > 27000 nM T57392 CD5J7W 50898619 IC50 = 10000 nM T57392 CU7TK4 50899749 IC50 > 20000 nM T57392 CZ9UD6 50901657 IC50 > 50000 nM T57392 C1N4YP 50908737 IC50 > 10000 nM T57392 CENW12 50925404 IC50 > 100000 nM T57392 CK1CD3 50925423 IC50 = 14300 nM T57392 CMF7T6 50925457 IC50 > 5000 nM T57392 C2GTE4 50938548 IC50 > 50000 nM T57392 C4DH0A 50938549 IC50 > 20000 nM T57392 CJ43IF 50941460 IC50 = 3000 nM T57392 CP7B9V 50942696 IC50 > 20000 nM T57392 CI32TR 50992246 IC50 > 25000 nM T57392 C2SHO8 50993865 IC50 = 2780 nM T57392 CNBU93 50994740 IC50 > 30000 nM T57392 CH82SZ 51000500 IC50 > 30000 nM T57392 CX48AD 51002362 IC50 > 45000 nM T57392 C4P8LX 51002580 IC50 = 14 nM T57392 CX6PZ9 51003130 IC50 = 3620 nM T57392 CAZQ43 51003133 IC50 = 11500 nM T57392 CQ8KP7 51003749 IC50 = 400 nM T57392 CP6NI2 51030711 IC50 > 30000 nM T57392 C70OGS 51030984 IC50 > 30000 nM T57392 CX28ZP 51030985 IC50 > 30000 nM T57392 CXB2Q6 51031001 IC50 > 30000 nM T57392 CUG03K 51033838 IC50 > 10000 nM T57392 C7OB2X 51035721 IC50 > 25000 nM T57392 C08FGN 51039225 IC50 = 5852 nM T57392 CS14BH 51039226 IC50 = 7957 nM T57392 CR70XF 51039227 IC50 = 4293 nM T57392 CA14XO 51051122 IC50 > 10000 nM T57392 C1RP3V 51051125 IC50 > 10000 nM T57392 C96AQN 51346908 IC50 > 30000 nM T57392 CGW84J 51346919 IC50 > 50000 nM T57392 C3I7XR 51346964 IC50 > 10000 nM T57392 C2IO7B 51346981 IC50 > 10000 nM T57392 CD2YU8 51351496 IC50 = 29000 nM T57392 C2UG4W 51351504 IC50 = 42000 nM T57392 CAO41L 51351511 IC50 > 30000 nM T57392 CG3PR6 52912222 IC50 > 33000 nM T57392 CJ86KR 52917690 IC50 > 20000 nM T57392 CUQ53T 52918018 IC50 = 1000 nM T57392 CTP6U5 52918019 IC50 = 340 nM T57392 CAXJ10 52918120 IC50 > 3162.28 nM T57392 CRN19G 52918121 IC50 > 3162.28 nM T57392 CTJ28K 52918135 IC50 > 50000 nM T57392 CJD25G 52920263 IC50 = 16000 nM T57392 C2RW5A 52940961 IC50 > 6000 nM T57392 CSXY62 52941059 IC50 = 30000 nM T57392 CQW15U 52941269 IC50 > 50000 nM T57392 C1YLX8 52941699 IC50 > 10000 nM T57392 C6NR7I 52942081 IC50 > 30000 nM T57392 C3BO1Z 52942119 IC50 = 30000 nM T57392 C34WMT 52942456 IC50 > 10000 nM T57392 C3TK2O 52943442 IC50 = 30000 nM T57392 CHD7O6 52943758 IC50 < 165 nM T57392 CTI28E 52944579 IC50 > 50000 nM T57392 CX0YD9 52944600 IC50 = 16600 nM T57392 CXTM57 52944645 IC50 > 30000 nM T57392 C4I6ML 52944843 IC50 = 200 nM T57392 CT6SQ3 52944941 IC50 = 3400 nM T57392 CO7ZR1 52947102 IC50 = 25000 nM T57392 C2YK4B 52947710 IC50 = 11600 nM T57392 C56NDZ 52948169 IC50 = 5900 nM T57392 C48JMX 52948255 IC50 > 50000 nM T57392 C7SAC6 52948857 IC50 > 10000000 nM T57392 C43KTX 52948925 IC50 = 11600 nM T57392 C4LVO6 52948971 IC50 = 400 nM T57392 C0HA6F 52949188 IC50 > 25000 nM T57392 C3DTV5 53233133 IC50 > 10000 nM T57392 C2RCZ0 53235503 IC50 > 20000 nM T57392 C9RIJ7 53237893 IC50 = 2800 nM T57392 C5ZT7N 53237897 IC50 = 500 nM T57392 C4KRV8 53237899 IC50 = 3300 nM T57392 C0H6TR 53237903 IC50 = 900 nM T57392 CIP64Q 53238125 IC50 = 1500 nM T57392 C8RV1B 53241150 IC50 = 900 nM T57392 CQIY23 53248846 IC50 > 50000 nM T57392 C9MHR0 53248847 IC50 > 50000 nM T57392 CG3LA9 53248849 IC50 = 230 nM T57392 CT9V3I 53251325 IC50 > 100000 nM T57392 CD35QU 53308640 IC50 > 10000 nM T57392 CRI92N 53311230 IC50 > 10000 nM T57392 CQ9HO5 53311701 IC50 = 20000 nM T57392 CL78NK 53316823 IC50 = 917 nM T57392 C1-MAY-02 53317017 IC50 > 50000 nM T57392 C7IMH5 53317594 IC50 > 10000 nM T57392 CT56HN 53317595 IC50 = 7533 nM T57392 CK27PC 53317643 IC50 = 50000 nM T57392 C9I3NE 53317658 IC50 > 10000 nM T57392 CXV3W2 53317718 IC50 > 50000 nM T57392 CP14EK 53317957 IC50 > 50000 nM T57392 CL45CT 53318503 IC50 > 5000 nM T57392 CDCA26 53318560 IC50 > 10000 nM T57392 C5F1IR 53318745 IC50 > 25000 nM T57392 CD0H8Z 53318872 IC50 = 3385 nM T57392 C90DGH 53318873 IC50 > 10000 nM T57392 C9MJ6C 53318874 IC50 = 10000 nM T57392 CZ0M8J 53319021 IC50 = 8 nM T57392 CJ2D3F 53319267 IC50 > 25000 nM T57392 COJ82D 53319320 IC50 > 50000 nM T57392 CK2G3D 53319480 IC50 = 154 nM T57392 C90TZS 53319482 IC50 = 57 nM T57392 CTA23R 53319654 IC50 = 50000 nM T57392 CXY8A4 53319905 IC50 > 38000 nM T57392 CWV40O 53320177 IC50 = 4346 nM T57392 CY5PO1 53320189 IC50 = 8845 nM T57392 CXF1S4 53320328 IC50 = 41 nM T57392 CB84NG 53320778 IC50 = 1160 nM T57392 C5HL4R 53321372 IC50 > 25000 nM T57392 C9JVY1 53321494 IC50 = 3093 nM T57392 CQ9PR5 53321511 IC50 = 7224 nM T57392 CW28NZ 53321512 IC50 = 6466 nM T57392 C4X3IS 53321979 IC50 = 4870 nM T57392 CLD82J 53322084 IC50 = 67 nM T57392 CY09UA 53322086 IC50 = 33 nM T57392 CBUT35 53322087 IC50 = 495 nM T57392 CMH54U 53322279 IC50 > 50000 nM T57392 C9JUC1 53322838 IC50 = 1427 nM T57392 CEH78Z 53322839 IC50 = 5684 nM T57392 C78CYN 53322959 IC50 = 2605 nM T57392 CR57HN 53323639 IC50 = 32000 nM T57392 CX54CT 53323813 IC50 = 8500 nM T57392 C01OZU 53324167 IC50 = 5707 nM T57392 CC08MY 53324265 IC50 = 36000 nM T57392 C0GIP4 53324272 IC50 > 10000 nM T57392 CC1ER2 53324598 IC50 > 30000 nM T57392 CW58QL 53324656 IC50 = 100 nM T57392 C3QNR2 53325463 IC50 = 1500 nM T57392 CZN8B4 53325581 IC50 = 20 nM T57392 C1WJH5 53325600 IC50 > 10000 nM T57392 CZ1SE0 53325908 IC50 > 50000 nM T57392 C1N7XO 53325966 IC50 = 6020 nM T57392 C28HNA 53326213 IC50 = 31000 nM T57392 C4VG5W 53326249 IC50 > 100000 nM T57392 CVNH56 53326712 IC50 = 973 nM T57392 C4ZUJ9 53326724 IC50 > 10000 nM T57392 CU05TQ 53326725 IC50 > 10000 nM T57392 C9Z3WY 53326726 IC50 = 4363 nM T57392 CE9NR7 53326727 IC50 = 9373 nM T57392 C18TPG 53326909 IC50 > 25000 nM T57392 C7J8ZY 53327611 IC50 > 30000 nM T57392 C8PJ6E 53354789 IC50 = 13000 nM T57392 CYMP74 53354793 IC50 = 40000 nM T57392 C8ZRE3 53356518 IC50 > 40000 nM T57392 CL89US 53359023 IC50 > 50000 nM T57392 CRZL59 53361076 IC50 > 40000 nM T57392 C9H5YE 53361128 IC50 > 10000 nM T57392 CC7DZ4 53362086 IC50 > 50000 nM T57392 CX83CK 53362097 IC50 > 8900 nM T57392 C1F8IK 53363810 IC50 > 30000 nM T57392 C9GYZ3 53372790 IC50 = 500 nM T57392 CT6K2O 53373472 IC50 = 4000 nM T57392 C9CT8N 53373573 IC50 = 6309.57 nM T57392 CL37YO 53380288 IC50 > 10000 nM T57392 C1Q0OJ 53382545 IC50 > 30000 nM T57392 C19HFO 53386426 IC50 = 16600 nM T57392 CZWO31 53387025 IC50 > 33300 nM T57392 C7KM5B 53388319 IC50 > 10000 nM T57392 CIGM78 53389570 IC50 > 30000 nM T57392 C5B1ST 53391517 IC50 = 560 nM T57392 CKOD62 53391618 IC50 = 2610 nM T57392 CD24UN 53391714 IC50 = 12800 nM T57392 CQ4E2W 53391716 IC50 = 13600 nM T57392 C64TJO 53391717 IC50 = 9420 nM T57392 C3Q6IL 53391718 IC50 = 10800 nM T57392 C6AYE3 53392451 IC50 > 33300 nM T57392 C0JI1M 53392850 IC50 < 50 nM T57392 C8K1TZ 53392852 IC50 < 50 nM T57392 C47VGW 53393916 IC50 = 7900 nM T57392 C24FQU 53465297 IC50 > 12000 nM T57392 C0T5VA 53467975 IC50 > 11000 nM T57392 C2XHO3 53468206 IC50 > 11000 nM T57392 CX0R1K 53469059 IC50 > 25000 nM T57392 CV7C0D 53469060 IC50 = 23700 nM T57392 CCKD45 53469061 IC50 > 25000 nM T57392 C3SRN7 53469411 IC50 > 40000 nM T57392 CK1C9O 53472113 IC50 = 7000 nM T57392 CITN21 53475321 IC50 > 20000 nM T57392 C9EF7S 53482945 IC50 = 15000 nM T57392 CFU8T7 53483937 IC50 > 30000 nM T57392 CG3FA9 53492750 IC50 > 50000 nM T57392 C4U5IX 53493001 IC50 > 35000 nM T57392 CE9K7U 53494972 IC50 > 10000 nM T57392 C7TR2W 53497131 IC50 > 30000 nM T57392 CGSN74 53497490 IC50 = 8700 nM T57392 CVA4I0 54576291 IC50 > 10000 nM T57392 CSAV94 54576503 IC50 > 10000 nM T57392 COF6B0 54577892 IC50 > 30000 nM T57392 C2ECL9 54577896 IC50 > 30000 nM T57392 CP24ZC 54579002 IC50 = 17900 nM T57392 C7FXV6 54580144 IC50 = 25000 nM T57392 C6R3MZ 54580973 IC50 = 230 nM T57392 C2XV8F 54581365 IC50 = 600 nM T57392 CQ0YA3 54581861 IC50 = 380 nM T57392 CWKA42 54582019 IC50 = 1260 nM T57392 CB8JV7 54582823 IC50 > 20000 nM T57392 CF5Q0W 54583932 IC50 = 300 nM T57392 CHP62C 54584119 IC50 = 16000 nM T57392 C37TZQ 54584868 IC50 > 30000 nM T57392 CY4F0W 54584873 IC50 = 1600 nM T57392 CQ0G6R 54586630 IC50 = 9000 nM T57392 CQWI92 54586805 IC50 > 30000 nM T57392 C8MH6B 54587759 IC50 > 20000 nM T57392 CXU62W 54677935 IC50 > 40000 nM T57392 C0ZG2V 54709839 IC50 > 100000 nM T57392 CO75TL 54712015 IC50 > 50000 nM T57392 CLT3Q8 54716246 IC50 > 100000 nM T57392 CMN1C6 54752118 IC50 > 10000 nM T57392 CZY7F9 54752621 IC50 = 950 nM T57392 C69EQM 54752774 IC50 > 10000 nM T57392 CD8YN4 54753626 IC50 > 30000 nM T57392 CL32AY 54753627 IC50 > 30000 nM T57392 CBO2L1 54761157 IC50 > 40000 nM T57392 C0Y9ZG 54761473 IC50 > 10000 nM T57392 CS23GM 54762055 IC50 > 40000 nM T57392 CPS5V6 54764158 IC50 > 30000 nM T57392 CU62DN 54764919 IC50 > 30000 nM T57392 C0T3KY 54765285 IC50 > 11000 nM T57392 CJ9B4P 54768039 IC50 > 10000 nM T57392 C79DVG 56589615 IC50 > 30000 nM T57392 C4S1HX 56589672 IC50 = 39700 nM T57392 C23NQS 56593147 IC50 > 20000 nM T57392 CXSQ19 56593712 IC50 = 63200 nM T57392 C4U6BD 56593857 IC50 > 100000 nM T57392 CHD79F 56594864 IC50 > 10000 nM T57392 CMQ2J3 56594865 IC50 > 10000 nM T57392 C6FE3Z 56594866 IC50 > 10000 nM T57392 CS3E5I 56594867 IC50 > 10000 nM T57392 C9ZF6B 56643412 IC50 > 25000 nM T57392 CQ18BI 56643478 IC50 = 400 nM T57392 CBJ4V8 56649677 IC50 > 20000 nM T57392 CPJ7D3 56658546 IC50 > 30000 nM T57392 C7AG6I 56658547 IC50 > 30000 nM T57392 C6W5UT 56658548 IC50 > 30000 nM T57392 CFT9V8 56659147 IC50 > 25000 nM T57392 CGID30 56659201 IC50 > 10000 nM T57392 CX31TJ 56661748 IC50 = 7500 nM T57392 C2QTH5 56662000 IC50 > 30000 nM T57392 CC1GK4 56665357 IC50 > 30000 nM T57392 CC9XR7 56669562 IC50 > 10000 nM T57392 CXE9A8 56669563 IC50 > 8000 nM T57392 CK9L4C 56672570 IC50 > 30000 nM T57392 CZP86D 56677285 IC50 > 30000 nM T57392 C7QW5F 56678507 IC50 > 10000 nM T57392 CW7QF9 56679101 IC50 > 30000 nM T57392 CUIB93 56679632 IC50 > 400000 nM T57392 CK73UC 56683046 IC50 > 6000 nM T57392 CJC19B 56683709 IC50 > 30000 nM T57392 CY3G8F 56834936 IC50 > 30000 nM T57392 CPN57V 56834986 IC50 > 10000 nM T57392 CY92VU 56835087 IC50 = 11000 nM T57392 C0JMA7 56835088 IC50 = 6600 nM T57392 CBOD63 56835089 IC50 = 655 nM T57392 CR7LS4 56835090 IC50 > 30000 nM T57392 C7G5IR 56835177 Ki = 1122018.45 nM T57392 C3IZU1 56835179 Ki = 707945.78 nM T57392 C70GHX 56835991 IC50 = 32000 nM T57392 CH2AY6 56838673 IC50 > 30000 nM T57392 C3OE8N 56838888 IC50 = 10000 nM T57392 CVYF04 56840671 IC50 > 10000 nM T57392 CR8KU2 56840672 IC50 > 10000 nM T57392 CKY51C 56847605 IC50 = 54000 nM T57392 CUY28J 56850524 IC50 > 50 nM T57392 CK0I6Q 56850525 IC50 > 50 nM T57392 C1U7XJ 56924869 IC50 > 30000 nM T57392 CZRQ14 56929159 IC50 = 54000 nM T57392 C9IVD0 56929216 IC50 > 10000 nM T57392 C90URY 56929249 IC50 = 54000 nM T57392 CZ25SN 56935695 IC50 > 10000 nM T57392 CPAU51 56943206 IC50 = 5000 nM T57392 CI04WC 56948248 IC50 = 800 nM T57392 CL16UQ 56949326 IC50 > 30000 nM T57392 C89PEN 56949822 IC50 > 10000 nM T57392 C1K8TD 56949966 IC50 > 10000 nM T57392 C5LJE8 56951456 IC50 > 27000 nM T57392 C6N0ZI 56951457 IC50 > 27000 nM T57392 CL90EM 56951458 IC50 > 27000 nM T57392 CWB5H7 56953768 IC50 = 19400 nM T57392 CS0HF1 56953769 IC50 = 2610 nM T57392 CPJ7X3 56953770 IC50 = 5330 nM T57392 CK7M6W 56953771 IC50 = 50000 nM T57392 CO96BR 56953896 IC50 = 29400 nM T57392 CJ0WM6 56953897 IC50 = 50000 nM T57392 C4UV1D 56953898 IC50 = 2050 nM T57392 CPKI96 56954010 IC50 = 410 nM T57392 C6Q8BZ 56954011 IC50 = 20 nM T57392 C5G4UX 56954012 IC50 = 10500 nM T57392 C8UQ2S 56954013 IC50 = 1500 nM T57392 CHQA53 56954137 IC50 = 120 nM T57392 CZGE53 56954138 IC50 = 50000 nM T57392 CGRC25 56954242 IC50 = 1184 nM T57392 CRT0Y2 56954243 IC50 = 663 nM T57392 CKN0Z8 56964577 IC50 > 25000 nM T57392 CS7U9L 56965952 IC50 > 10000 nM T57392 CT67IO 57325589 IC50 > 25000 nM T57392 CV5CP4 57326678 IC50 = 8500 nM T57392 CQT5I3 57328465 IC50 > 27000 nM T57392 CW8B4D 57330208 IC50 > 27000 nM T57392 CLB5K0 57331386 IC50 > 10000 nM T57392 CGUA26 57331668 IC50 > 50000 nM T57392 CL45WN 57345320 IC50 = 320 nM T57392 CHE2I1 57345500 IC50 = 240 nM T57392 C63TFM 57345501 IC50 = 80 nM T57392 C8KT2F 57345502 IC50 = 160 nM T57392 C8CGX9 57345520 IC50 > 40000 nM T57392 CT8VZ6 57345658 IC50 > 30000 nM T57392 C7O0AI 57345659 IC50 > 30000 nM T57392 C3L9ZA 57345660 IC50 > 30000 nM T57392 CZK3M1 57345661 IC50 > 30000 nM T57392 C34DJP 57384236 IC50 > 50000 nM T57392 CEOC15 57384237 IC50 > 50000 nM T57392 CY50WC 57384238 IC50 > 50000 nM T57392 C7S0ZR 57384239 IC50 > 50000 nM T57392 C2XN1G 57384481 IC50 > 50000 nM T57392 CR73IZ 57384482 IC50 > 50000 nM T57392 CR2M5H 57384483 IC50 = 2700 nM T57392 CQ72HI 57384749 IC50 > 50000 nM T57392 C68KGE 57384750 IC50 > 50000 nM T57392 CCT5D4 57386783 IC50 > 50000 nM T57392 CC30XZ 57386784 IC50 > 50000 nM T57392 C79BXP 57386785 IC50 > 50000 nM T57392 CM6DV7 57387028 IC50 > 50000 nM T57392 C0GS4F 57387282 IC50 > 50000 nM T57392 C0TL9C 57387283 IC50 > 50000 nM T57392 CRV2P5 57387539 IC50 > 50000 nM T57392 CAU3G9 57387540 IC50 > 50000 nM T57392 CL2AO8 57387541 IC50 > 50000 nM T57392 C0XWL8 57387542 IC50 > 50000 nM T57392 CC4DK0 57387775 IC50 > 50000 nM T57392 C56ORS 57388650 IC50 > 10000 nM T57392 CMDX46 57390296 IC50 < 500 nM T57392 COYC39 57390989 IC50 > 25000 nM T57392 C5OJP0 57391102 IC50 > 25000 nM T57392 CR8MW2 57391205 IC50 > 10000 nM T57392 C6SGK0 57391843 IC50 > 20000 nM T57392 CL2C3I 57392070 IC50 < 500 nM T57392 CX7L1C 57392134 IC50 < 500 nM T57392 CT20WV 57392770 IC50 > 25000 nM T57392 C82KEB 57392771 IC50 = 1400 nM T57392 CNM1H3 57392772 IC50 = 12400 nM T57392 C07SCG 57392773 IC50 = 7000 nM T57392 CNQ9B2 57392969 IC50 > 10000 nM T57392 CHU04N 57393566 IC50 = 6900 nM T57392 CVO5M3 57393573 IC50 = 8700 nM T57392 C5IM8F 57393826 IC50 < 500 nM T57392 CHET54 57393827 IC50 < 500 nM T57392 CJ0V4M 57394499 IC50 > 20000 nM T57392 CVA02G 57394500 IC50 > 20000 nM T57392 C04IST 57394707 IC50 > 10000 nM T57392 CNOH63 57394711 IC50 > 10000 nM T57392 CSO4Z0 57395278 IC50 = 2500 nM T57392 C01VOH 57395286 IC50 = 2400 nM T57392 CB09IO 57395287 IC50 = 28300 nM T57392 C0BP8I 57396250 IC50 > 50000 nM T57392 C3DB0F 57396251 IC50 > 25000 nM T57392 C6HBG0 57396813 IC50 > 30000 nM T57392 CYC1Q5 57397055 IC50 = 18800 nM T57392 C25FTZ 57397056 IC50 = 15000 nM T57392 CJIZ48 57397373 IC50 < 500 nM T57392 CU4FW8 57397383 IC50 > 25000 nM T57392 CH32BO 57397434 IC50 < 500 nM T57392 CO14BW 57397444 IC50 < 500 nM T57392 CQS0M5 57397654 IC50 > 30000 nM T57392 C5D0RB 57398829 IC50 = 1900 nM T57392 CL4I6O 57398830 IC50 = 4400 nM T57392 CVRD17 57399109 IC50 < 500 nM T57392 CZLD01 57399119 IC50 < 500 nM T57392 CW2DO9 57399120 IC50 < 500 nM T57392 CK4BW0 57399710 IC50 = 780 nM T57392 C0OZM1 57399711 IC50 > 20000 nM T57392 C5BW8L 57399712 IC50 = 1900 nM T57392 CEC78U 57399713 IC50 > 20000 nM T57392 C5SJC7 57399714 IC50 > 20000 nM T57392 CE82XL 57400502 IC50 = 4900 nM T57392 CWZ50O 57400503 IC50 = 3600 nM T57392 C5MG6Q 57400504 IC50 = 15100 nM T57392 CJBU02 57400505 IC50 = 3300 nM T57392 CG7NW9 57400793 IC50 < 200 nM T57392 CR6AE3 57400851 IC50 < 500 nM T57392 CO1J9V 57401476 IC50 = 2900 nM T57392 C0MKN9 57402230 IC50 = 7000 nM T57392 C9D3ZE 57402314 IC50 = 1400 nM T57392 CXT2L1 57402315 IC50 > 20000 nM T57392 CYVN84 57402550 IC50 < 500 nM T57392 C5XF1Z 57402551 IC50 < 500 nM T57392 CTD73Q 57403212 IC50 > 50000 nM T57392 C4RHF3 57404027 IC50 > 30000 nM T57392 C9SB1D 57404031 IC50 = 18100 nM T57392 CKU6E8 57404500 IC50 > 30000 nM T57392 C6XA7G 57405264 IC50 > 30000 nM T57392 CUOV05 57411066 IC50 > 30000 nM T57392 C37SMZ 57505249 IC50 > 100000 nM T57392 C7I4QD 57519510 IC50 > 50000 nM T57392 C3N4MF 57520842 IC50 > 50000 nM T57392 CEL56T 57520942 IC50 > 50000 nM T57392 CAQ71K 57574919 IC50 > 20000 nM T57392 CASM07 57574933 IC50 > 20000 nM T57392 CM1EK8 57574953 IC50 > 20000 nM T57392 CX4F6L 57574973 IC50 > 20000 nM T57392 CY5D1K 57574980 IC50 > 20000 nM T57392 C9CD2Y 57574990 IC50 > 20000 nM T57392 C3XGL6 57574995 IC50 > 20000 nM T57392 CR7K1C 57575007 IC50 > 20000 nM T57392 CG93BU 57575012 IC50 > 20000 nM T57392 CPE25J 57575026 IC50 > 20000 nM T57392 CB30PQ 57656715 IC50 = 3100 nM T57392 CV2J9A 57663655 IC50 > 100000 nM T57392 CTM6K5 57690900 IC50 > 20000 nM T57392 C35GXV 57720515 EC50 > 40000 nM T57392 C58TKU 57773771 IC50 = 8100 nM T57392 C8I2JX 57798425 IC50 = 18000 nM T57392 C52UJG 57798468 IC50 = 4500 nM T57392 C0JCN7 57798480 IC50 = 26600 nM T57392 CLYT61 57798492 IC50 = 16000 nM T57392 CO7C9R 57798603 IC50 = 6900 nM T57392 C0VU2Z 57798682 IC50 > 50000 nM T57392 C1QX8T 57798887 IC50 = 32400 nM T57392 CO1B7C 57869916 IC50 = 27000 nM T57392 C9OBT1 57869953 IC50 > 50000 nM T57392 CD9XV0 57869954 IC50 > 50000 nM T57392 C4R6NA 57870014 IC50 = 24000 nM T57392 C2H8ZW 57870102 IC50 > 50000 nM T57392 C7C4VE 57870158 IC50 = 40000 nM T57392 C2CR3O 57870171 IC50 = 7600 nM T57392 C0QFL3 57877765 IC50 = 22100 nM T57392 CANZ90 57994936 IC50 > 20000 nM T57392 CGBY54 58063225 IC50 > 10000 nM T57392 C0P8VW 58063334 IC50 > 10000 nM T57392 CZO2J1 58063487 IC50 > 10000 nM T57392 C9JCL7 58080768 IC50 = 2900 nM T57392 CSC1K6 58109236 IC50 > 50000 nM T57392 CS05MK 58109240 IC50 > 50000 nM T57392 CDC28F 58109250 IC50 > 50000 nM T57392 C4E2RC 58109371 IC50 > 50000 nM T57392 C4SC0Z 58109674 IC50 > 50000 nM T57392 C1EF0B 58109729 IC50 > 50000 nM T57392 CBZX94 58199027 IC50 > 30000 nM T57392 CB72QI 58204997 IC50 > 10000 nM T57392 C93STQ 58239274 IC50 > 20000 nM T57392 C2SE1Z 58239287 IC50 > 20000 nM T57392 CI45ZP 58269513 IC50 > 30000 nM T57392 CK10DA 58269516 IC50 > 30000 nM T57392 CV9FC4 58269518 IC50 > 30000 nM T57392 CM1GN4 58269523 IC50 > 30000 nM T57392 CAY0H7 58269562 IC50 > 30000 nM T57392 CN13SI 58269563 IC50 > 30000 nM T57392 CPQ0Z4 58269588 IC50 > 30000 nM T57392 C8A3JQ 58269598 IC50 > 30000 nM T57392 CD18IU 58269609 IC50 > 30000 nM T57392 CQV75S 58269620 IC50 = 12000 nM T57392 C26OPT 58269625 IC50 > 30000 nM T57392 C8ILS3 58269629 IC50 > 30000 nM T57392 C5VFQ7 58269655 IC50 > 30000 nM T57392 CQ63WZ 58269663 IC50 > 30000 nM T57392 C2PYB1 58269668 IC50 > 30000 nM T57392 CI3P0D 58269670 IC50 = 27000 nM T57392 C5RF8T 58269685 IC50 = 10000 nM T57392 C4OS3J 58269689 IC50 = 11000 nM T57392 C3CFB8 58269691 IC50 > 30000 nM T57392 CZ71SN 58282592 IC50 = 40 nM T57392 CZA32V 58344912 IC50 > 10000 nM T57392 CPVF85 58344916 IC50 > 10000 nM T57392 CY62SG 58345029 IC50 > 10000 nM T57392 CJ68YT 58393461 IC50 = 1500 nM T57392 CY9I6G 58393477 IC50 < 300 nM T57392 CAI83V 58393493 IC50 = 2400 nM T57392 C65ORN 58393495 IC50 = 2500 nM T57392 C4COR1 58393517 IC50 < 300 nM T57392 CNW5T4 58393622 IC50 > 10000 nM T57392 CY6F0D 58393650 IC50 < 300 nM T57392 C0J6DV 58393772 IC50 < 300 nM T57392 CF7U6N 58393782 IC50 > 10000 nM T57392 CUKP69 58393851 IC50 < 300 nM T57392 CVW3J5 58393864 IC50 < 300 nM T57392 CG50XR 58393885 IC50 = 9500 nM T57392 CC7LE9 58393895 IC50 < 300 nM T57392 COD27G 58393915 IC50 < 300 nM T57392 CJ9P7S 58393925 IC50 = 730 nM T57392 C84USG 58393938 IC50 < 300 nM T57392 CB6Y9V 58393939 IC50 < 300 nM T57392 CHPD56 58393945 IC50 < 300 nM T57392 C54QRX 58394136 IC50 > 10000 nM T57392 CYW78T 58394137 IC50 < 300 nM T57392 C0F3BO 58394783 IC50 > 10000 nM T57392 C0X7IK 58394837 IC50 > 10000 nM T57392 CASI81 58395078 IC50 > 10000 nM T57392 CWBM72 58395283 IC50 > 10000 nM T57392 C6BZ0G 58439416 IC50 > 30000 nM T57392 C35FWX 58486367 IC50 > 10000 nM T57392 CJV84Q 58534983 IC50 > 10000 nM T57392 C6JKM0 58834906 IC50 > 100000 nM T57392 CF9Z0L 58834953 IC50 > 26000 nM T57392 C4PWA9 58835024 IC50 > 40000 nM T57392 CCR4T7 58835217 IC50 > 73000 nM T57392 C5UJ4T 58863082 IC50 > 30000 nM T57392 CNM1V0 58863113 IC50 > 30000 nM T57392 C5FOK7 58863126 IC50 > 30000 nM T57392 CU89KE 58863146 IC50 > 30000 nM T57392 CNE1Q4 58863165 IC50 > 30000 nM T57392 CM58WY 58863171 IC50 > 30000 nM T57392 CO4NR9 58863217 IC50 > 30000 nM T57392 CK5P3B 58863232 IC50 > 30000 nM T57392 C9ZE7J 58874273 IC50 > 50000 nM T57392 C7CE6L 58950132 IC50 = 17900 nM T57392 CCQM76 59153288 IC50 > 50000 nM T57392 C3L4JY 59176329 IC50 > 10000 nM T57392 CMK4G5 59177101 IC50 = 230 nM T57392 C0U1HA 59179260 IC50 > 10000 nM T57392 CK7T6D 59179887 IC50 > 10000 nM T57392 C6DG2S 59190464 IC50 > 1000 nM T57392 CL9R5M 59190503 IC50 > 1000 nM T57392 C79GHB 59190548 IC50 > 1000 nM T57392 CJ6R8Q 59251679 IC50 > 25000 nM T57392 C2PJ4N 59271992 IC50 > 20000 nM T57392 CUE79I 59272004 IC50 > 10000 nM T57392 C19YVT 59377518 IC50 > 32000 nM T57392 C1JK7V 59377559 IC50 > 50000 nM T57392 C0Q2OB 59396176 IC50 = 3700 nM T57392 C67THA 59396210 IC50 = 1300 nM T57392 CZVU58 59396246 IC50 < 390 nM T57392 CDA17U 59396249 IC50 = 780 nM T57392 CNA14Q 59396273 IC50 < 780 nM T57392 C40NHU 59396275 IC50 = 1300 nM T57392 CM67CI 59396283 IC50 = 1600 nM T57392 CD7UI0 59396290 IC50 = 30200 nM T57392 CF3EX0 59396298 IC50 = 5600 nM T57392 CE72HG 59396348 IC50 < 780 nM T57392 CV9I1W 59396356 IC50 < 300 nM T57392 CI56OZ 59396371 IC50 = 17900 nM T57392 CK9C2P 59396429 IC50 < 780 nM T57392 CT5CQ2 59396449 IC50 = 1400 nM T57392 CE7JV9 59396534 IC50 < 390 nM T57392 CXP57T 59396609 IC50 = 1600 nM T57392 CZ6FR9 59396619 IC50 < 390 nM T57392 C4GF0P 59396624 IC50 = 1000 nM T57392 CFDG19 59401765 IC50 > 30000 nM T57392 CC5QW1 59401793 IC50 > 30000 nM T57392 CNOI48 59401886 IC50 > 30000 nM T57392 CJ2Y3A 59414201 IC50 = 3100 nM T57392 CVZ09Q 59454159 IC50 = 700 nM T57392 CK6LX0 59454220 IC50 = 9000 nM T57392 C2SDN1 59454252 IC50 = 32000 nM T57392 CK6W7I 59536635 IC50 > 10000 nM T57392 CA9NE4 59548712 IC50 > 30000 nM T57392 CM1G2P 59568656 IC50 > 50000 nM T57392 CP2UY3 59634686 IC50 > 27000 nM T57392 CPA0L2 59634709 IC50 > 27000 nM T57392 CS80HW 59648012 IC50 > 30000 nM T57392 C3RB0E 59648133 IC50 > 50000 nM T57392 CYKF93 59651916 IC50 > 30000 nM T57392 C5PDB3 59651957 IC50 > 30000 nM T57392 C4W8RH 59651989 IC50 > 30000 nM T57392 CBEG02 59721267 IC50 = 6500 nM T57392 CV6L5Y 59721273 IC50 = 1300 nM T57392 CS5U7D 59721308 IC50 = 800 nM T57392 CK2UR9 59721409 IC50 = 600 nM T57392 C4I3JA 59721419 IC50 = 400 nM T57392 C7ECU2 59794447 IC50 > 40000 nM T57392 C1MVB2 59835725 IC50 > 50000 nM T57392 CZ6EF7 59835728 IC50 > 10000 nM T57392 CMG1L8 59835758 IC50 > 50000 nM T57392 C42PAO 59835879 IC50 > 50000 nM T57392 C2W1TF 60001863 IC50 = 47400 nM T57392 CK5N4E 60148693 IC50 = 2700 nM T57392 C6L4RH 60148695 IC50 > 45000 nM T57392 CUYB59 60148924 IC50 = 12800 nM T57392 C4MV2N 60149678 IC50 = 18000 nM T57392 CTL97W 60151476 IC50 > 45000 nM T57392 C62SQG 60155628 IC50 > 20000 nM T57392 COS39T 60155629 IC50 > 10000 nM T57392 CE5A7B 60162406 IC50 > 40000 nM T57392 C2D3HQ 60168069 IC50 > 30000 nM T57392 CIJ16Y 60196616 IC50 > 30000 nM T57392 C3S1RP 60197614 IC50 > 30000 nM T57392 CS4F2O 60197712 IC50 > 30000 nM T57392 C87HTO 60197713 IC50 > 30000 nM T57392 C5ES4W 60197714 IC50 > 30000 nM T57392 CF19XN 60197716 IC50 > 30000 nM T57392 COI61M 60197822 IC50 > 30000 nM T57392 CP1CK0 60197823 IC50 > 30000 nM T57392 C0JL3I 60197824 IC50 > 30000 nM T57392 CVOF90 60197825 IC50 > 30000 nM T57392 CBN3G4 60197937 IC50 > 30000 nM T57392 CT26JV 60202329 IC50 > 50000 nM T57392 CWA0B6 60204017 IC50 > 30000 nM T57392 CW3H0V 60634975 IC50 = 10000 nM T57392 C4BZ2N 60637368 IC50 < 10000 nM T57392 C9F4JW 62705832 IC50 < 2500 nM T57392 CJ5HI6 66547425 IC50 < 1000 nM T57392 CH76RD 66550504 IC50 > 25000 nM T57392 C2LBW7 66551925 IC50 > 50000 nM T57392 CLHX28 66553128 IC50 > 20000 nM T57392 CNDH38 66557868 IC50 > 10000 nM T57392 CUC7B3 66557964 IC50 > 30000 nM T57392 C1LB6D 66558197 IC50 = 88000 nM T57392 C7UKS4 66558379 IC50 = 208000 nM T57392 CCK6E5 66558639 IC50 = 10000 nM T57392 C23NWU 66562843 IC50 > 20000 nM T57392 CE2S6P 66562938 IC50 > 20000 nM T57392 CK9FO4 66562947 IC50 > 20000 nM T57392 C1WXS5 66563037 IC50 > 20000 nM T57392 CG34JD 66563137 IC50 > 20000 nM T57392 C6LVU1 66563478 IC50 > 20000 nM T57392 C7FX5M 66563570 IC50 > 20000 nM T57392 C24BOR 66563571 IC50 > 20000 nM T57392 CQY3J2 66563572 IC50 > 20000 nM T57392 CY81CB 66575661 IC50 > 20000 nM T57392 CMXA10 66575743 IC50 > 50000 nM T57392 CZF76R 66608383 IC50 > 30000 nM T57392 CS72TK 66610926 IC50 > 10000 nM T57392 CVB4T1 66611375 IC50 > 10000 nM T57392 CUP41L 66613450 IC50 >= 30000 nM T57392 CFI5T8 66613669 IC50 > 10000 nM T57392 CY9TD4 66730677 IC50 > 10000 nM T57392 CJFS84 66731186 IC50 > 10000 nM T57392 CG1O8H 66734740 IC50 > 10000 nM T57392 C8CLK2 66735127 IC50 > 10000 nM T57392 CL5GH9 66735487 IC50 > 10000 nM T57392 CKN2U0 66764813 IC50 > 30000 nM T57392 CF15KL 66771109 IC50 = 15000 nM T57392 C51XCV 66781377 IC50 = 5880 nM T57392 CU6E0A 66818541 IC50 > 30000 nM T57392 CKD8I1 66818569 IC50 > 30000 nM T57392 C5LU1Z 66818766 IC50 > 30000 nM T57392 C5J4MR 66850717 IC50 > 10000 nM T57392 C40FKD 66898172 IC50 > 50000 nM T57392 C7TJ9X 66898814 IC50 > 50000 nM T57392 CX1P8I 67042254 IC50 > 25000 nM T57392 CFM6H7 67049587 IC50 > 100000 nM T57392 C4NX6W 67070065 IC50 > 50000 nM T57392 CN8AS7 67072266 IC50 = 170000 nM T57392 CVT35R 67097557 IC50 > 50000 nM T57392 CSQ3J1 67098421 IC50 = 2000 nM T57392 CJV8O4 67098558 IC50 > 50000 nM T57392 CE49GC 67098566 IC50 > 50000 nM T57392 COD28B 67098794 IC50 = 46000 nM T57392 C23QPJ 67098846 IC50 = 7700 nM T57392 C13OVI 67098869 IC50 = 29000 nM T57392 C9KQT3 67098926 IC50 = 7200 nM T57392 C52XBW 67098971 IC50 = 6500 nM T57392 CY76UR 67305743 IC50 = 15000 nM T57392 CQ70DL 67311221 IC50 = 5100 nM T57392 C3UKG8 67312397 IC50 = 1000 nM T57392 CM6TZ3 67312506 IC50 = 11000 nM T57392 CKMV48 67345882 IC50 > 10000 nM T57392 C50IMJ 67387021 IC50 > 20000 nM T57392 C4R8OG 67401728 IC50 > 30000 nM T57392 CX8JP5 67402849 IC50 > 40000 nM T57392 CPV39L 67406727 IC50 > 30000 nM T57392 C4S3FE 67450880 IC50 = 54000 nM T57392 C8L5HO 67453320 IC50 > 100000 nM T57392 C37YHJ 67496729 IC50 > 30000 nM T57392 C6QVG9 67538612 IC50 < 780 nM T57392 CNB15W 67607112 IC50 > 10000 nM T57392 CHU12R 67950044 IC50 > 10000 nM T57392 CDH49P 67950241 IC50 = 1100 nM T57392 CE94JQ 67953283 IC50 > 50000 nM T57392 CT43SM 67953330 IC50 > 50000 nM T57392 CPTA39 67953837 IC50 = 18000 nM T57392 CBO8G1 67971622 IC50 = 420 nM T57392 CV7BH5 67971878 IC50 = 4500 nM T57392 C5K7QG 67974411 IC50 >= 30000 nM T57392 CO75NL 68011817 IC50 > 10000 nM T57392 C02LWX 68074963 IC50 = 10000 nM T57392 CGW5L9 68075088 IC50 = 3000 nM T57392 CN3KZ8 68161075 IC50 = 8000 nM T57392 C32TVX 68230798 IC50 > 10000 nM T57392 C5YCB6 68234668 IC50 > 40000 nM T57392 CR17ZU 68234693 IC50 > 40000 nM T57392 CZCP37 68234870 IC50 > 100000 nM T57392 C9J8GY 68234878 IC50 > 40000 nM T57392 CN6KL0 68235029 IC50 > 40000 nM T57392 C1KAG4 68235232 IC50 > 40000 nM T57392 C68RYQ 68269759 IC50 = 5000 nM T57392 C7TR4I 68276577 IC50 > 10000 nM T57392 CK5V3O 68277611 IC50 > 10000 nM T57392 C17JAZ 68284084 IC50 > 30000 nM T57392 CCT07V 68290289 IC50 > 20000 nM T57392 C4LKB3 68291752 IC50 > 20000 nM T57392 CMG58Q 68295585 IC50 > 10000 nM T57392 CPA95O 68380152 IC50 > 30000 nM T57392 C95VPL 68380260 IC50 > 30000 nM T57392 CVM9Q1 68503758 IC50 > 50000 nM T57392 CJ2F6B 68506266 IC50 = 43000 nM T57392 C20LBF 68509511 IC50 = 19000 nM T57392 C1XL6P 68511915 IC50 = 4200 nM T57392 C5JYB8 68515257 IC50 > 20000 nM T57392 C69OHY 68560854 IC50 = 40000 nM T57392 CCD89X 68563058 IC50 = 3000 nM T57392 C48EIQ 68568011 IC50 > 100000 nM T57392 C0MYB6 68653619 IC50 > 20000 nM T57392 CH3Z7F 68658979 IC50 > 70000 nM T57392 C89CQS 68779277 IC50 > 10000 nM T57392 CJVI10 68882695 IC50 = 32300 nM T57392 CN0MY2 68994312 IC50 < 1000 nM T57392 CCIV97 68995742 IC50 < 1000 nM T57392 C17BRZ 68997664 IC50 < 1000 nM T57392 CJI32G 69081964 IC50 > 30000 nM T57392 CPGC67 69285465 IC50 > 40000 nM T57392 CM5XA1 69285531 IC50 = 20000 nM T57392 C0QZ4U 69285563 IC50 > 40000 nM T57392 C5T2GC 69285794 IC50 = 320 nM T57392 C8R4LZ 69286108 IC50 = 730 nM T57392 CNT95I 69286635 IC50 = 10 nM T57392 COJ4Q1 69315206 IC50 > 50000 nM T57392 CJ5Z7T 69316129 IC50 > 50000 nM T57392 C5VJG4 69643233 IC50 > 30000 nM T57392 CHD80I 69937162 IC50 > 50000 nM T57392 CAR2N8 69937236 IC50 > 50000 nM T57392 CN7X0U 69937257 IC50 > 50000 nM T57392 CC8QU9 70227534 IC50 > 10000 nM T57392 C06WFN 70276830 IC50 > 31622.78 nM T57392 CDQ85E 70276990 IC50 = 630.96 nM T57392 CK26FY 70295607 IC50 > 10000 nM T57392 CV4X5S 70295927 IC50 = 4500 nM T57392 CXD5V6 70297609 IC50 = 10000 nM T57392 CK5H1Y 70497007 IC50 > 10000 nM T57392 C6NSG3 70497750 IC50 > 10000 nM T57392 CWP52K 70497865 IC50 > 10000 nM T57392 C7VJ6A 70647728 IC50 > 40000 nM T57392 CAR46Z 70675172 IC50 > 25000 nM T57392 C97WSO 70678458 IC50 > 30000 nM T57392 CC6T5K 70679283 IC50 > 30000 nM T57392 C7W3JA 70681326 IC50 > 5000 nM T57392 C8XC1S 70682487 IC50 > 20000 nM T57392 CPF92N 70682528 IC50 = 16000 nM T57392 C37CFL 70682529 IC50 > 20000 nM T57392 CT94WJ 70684556 IC50 > 30000 nM T57392 CZHB48 70684601 IC50 = 15000 nM T57392 C5P0CI 70684602 IC50 = 20000 nM T57392 C86ETQ 70684603 IC50 > 20000 nM T57392 CCM9Z5 70684604 IC50 > 20000 nM T57392 C4FH7S 70684606 IC50 > 20000 nM T57392 CHFM92 70685176 IC50 = 5000 nM T57392 CG6BY1 70685177 IC50 = 5000 nM T57392 CWIC42 70685308 IC50 > 10000 nM T57392 C60SBP 70685515 IC50 = 4000 nM T57392 C3UO2F 70686000 IC50 = 5140 nM T57392 CYO5N3 70686766 IC50 >= 5000 nM T57392 C4VU7J 70688210 IC50 > 50000 nM T57392 CVFM91 70688283 IC50 > 200000 nM T57392 CZC4Y2 70688845 IC50 > 20000 nM T57392 CE1GI4 70688847 IC50 > 20000 nM T57392 C18OFS 70688848 IC50 > 20000 nM T57392 C4GXP2 70690453 IC50 > 30000 nM T57392 CJYB28 70691043 Ki = 520 nM T57392 C0XRC9 70691981 IC50 > 8600 nM T57392 CJ0P9G 70693067 IC50 > 20000 nM T57392 C8IOC9 70693068 IC50 = 15000 nM T57392 CF5YQ9 70693069 IC50 = 14000 nM T57392 CI4KP9 70693070 IC50 > 20000 nM T57392 CG4S9N 70693071 IC50 = 20000 nM T57392 CZT8D2 70693181 Ki = 3500 nM T57392 C6P3XM 70693710 IC50 = 340 nM T57392 C8G4AV 70694560 IC50 > 100000 nM T57392 CC6GZ9 70695067 IC50 > 20000 nM T57392 C75YPE 70695115 IC50 >= 5000 nM T57392 CS1MU4 70695116 IC50 > 20000 nM T57392 C6K9BL 70695117 IC50 = 15000 nM T57392 C1YZ6K 70695118 IC50 > 20000 nM T57392 C53RQN 70695119 IC50 = 18000 nM T57392 CXJ5V2 70695120 IC50 = 18000 nM T57392 CCR12A 70695121 IC50 > 20000 nM T57392 CVU08A 70695812 IC50 > 25000 nM T57392 CT1GF8 70697151 IC50 >= 5000 nM T57392 CSX71G 70697153 IC50 > 20000 nM T57392 C4JY5R 70697154 IC50 > 20000 nM T57392 CT78JN 70697155 IC50 > 20000 nM T57392 C34WHG 70697225 IC50 < 100 nM T57392 CBDL19 70792359 IC50 > 100000 nM T57392 C7DO1N 70817239 IC50 > 20000 nM T57392 C6L7FH 70817382 IC50 > 20000 nM T57392 C2PJ1D 70865101 IC50 > 30000 nM T57392 CUCQ24 70874317 IC50 = 20000 nM T57392 C8LCK6 70874412 IC50 = 4700 nM T57392 C1H7VK 70874453 IC50 = 2000 nM T57392 CJF91M 70874544 IC50 = 5700 nM T57392 C9EWB8 70874603 IC50 = 95000 nM T57392 C82PUD 70874605 IC50 = 19500 nM T57392 C8Q4LJ 70874786 IC50 = 4800 nM T57392 CF1G3K 70874916 IC50 > 100000 nM T57392 C30AJI 70914208 IC50 = 1400 nM T57392 C71AZM 70914219 IC50 = 40000 nM T57392 C2TC8W 70914230 IC50 = 38000 nM T57392 C8V5NF 70914234 IC50 = 94000 nM T57392 CP8HI7 70914358 IC50 = 152000 nM T57392 C3JKG2 70960031 IC50 = 66400 nM T57392 CXW7U0 70977933 IC50 > 10000 nM T57392 C1VMF2 70977969 IC50 > 50000 nM T57392 CA6GI0 70993878 IC50 = 1300 nM T57392 CGXQ60 71041800 IC50 = 600 nM T57392 C3J4SN 71041846 IC50 = 5700 nM T57392 C2HGI7 71153408 IC50 > 10000 nM T57392 C62ULC 71225056 IC50 > 100000 nM T57392 C7Y2LB 71230234 IC50 > 10000 nM T57392 C5RE4T 71244643 IC50 > 10000 nM T57392 C6BE5X 71271461 IC50 > 50000 nM T57392 CYLA18 71279311 IC50 = 3000 nM T57392 C2YHK4 71279453 IC50 > 8000 nM T57392 CKJ58I 71279693 IC50 = 19000 nM T57392 C7KQZ0 71279846 IC50 = 12000 nM T57392 C61BWN 71280407 IC50 = 5000 nM T57392 C63EIL 71280539 IC50 = 11000 nM T57392 CUP25C 71280634 IC50 = 48000 nM T57392 C4AP9F 71288434 IC50 = 12000 nM T57392 CAO07V 71293843 IC50 > 40000 nM T57392 CWN2M1 71300316 IC50 > 30000 nM T57392 C03KNO 71300317 IC50 > 30000 nM T57392 CWY4S0 71304814 IC50 > 50000 nM T57392 CS9OV5 71315139 IC50 = 71000 nM T57392 CR37DA 71419478 IC50 = 316.23 nM T57392 C5SML3 71449452 IC50 = 316.23 nM T57392 CL6BC1 71449606 IC50 = 72000 nM T57392 CDI84E 71450922 IC50 > 30000 nM T57392 CCL8I2 71451192 IC50 = 40000000 nM T57392 CCR9W0 71451887 IC50 = 27000 nM T57392 COQ0P1 71453071 IC50 = 199.53 nM T57392 C47GYB 71454279 IC50 > 10000 nM T57392 CJM13D 71454747 IC50 = 33000000 nM T57392 C0YD9K 71455398 IC50 = 2000 nM T57392 CR9VU6 71455427 IC50 = 6000 nM T57392 C4O2GZ 71457203 IC50 = 19700 nM T57392 C7MNB5 71457264 IC50 = 14700 nM T57392 C6X1GN 71457767 IC50 = 480 nM T57392 C3BF5T 71459944 IC50 = 21000 nM T57392 CD81EJ 71463058 IC50 = 1300 nM T57392 C0GBL7 71466345 IC50 > 20000 nM T57392 C3G9YK 71494647 IC50 = 14500 nM T57392 C8U0TA 71510812 IC50 > 25000 nM T57392 C9DIK2 71512060 IC50 > 10000 nM T57392 CF05BU 71513157 IC50 > 10000 nM T57392 CS1ZX0 71513822 IC50 > 10000 nM T57392 C0VLE3 71516457 IC50 > 20000 nM T57392 C2LVY0 71516458 IC50 > 20000 nM T57392 C1N2HF 71517046 IC50 = 8000 nM T57392 C7GS4P 71517047 IC50 = 3400 nM T57392 CWLO57 71517048 IC50 = 1600 nM T57392 C87CZW 71517049 IC50 > 20000 nM T57392 CY0VJ8 71517192 IC50 = 1000 nM T57392 C5S0XY 71517194 IC50 = 2600 nM T57392 C31DLT 71517195 IC50 = 8300 nM T57392 CRG0P7 71517196 IC50 = 14000 nM T57392 CA07TC 71517197 IC50 = 13000 nM T57392 CZ03XO 71519496 IC50 > 20000 nM T57392 C3CT1R 71530223 IC50 > 10000 nM T57392 CN8CM1 71533722 IC50 > 100000 nM T57392 C67ZSQ 71540073 IC50 > 30000 nM T57392 CE8YO0 71541095 IC50 = 2300 nM T57392 CN79ZY 71541096 IC50 > 20000 nM T57392 CNCR14 71541097 IC50 = 3900 nM T57392 CW34SU 71541098 IC50 = 10200 nM T57392 CKW24J 71541099 IC50 = 7600 nM T57392 C0ZL6O 71541186 IC50 = 11000 nM T57392 C92PZK 71541187 IC50 = 18000 nM T57392 C0T4RD 71541188 IC50 = 6700 nM T57392 CB91FO 71541189 IC50 = 5100 nM T57392 CY5E0J 71541190 IC50 = 3900 nM T57392 C4XK1S 71541191 IC50 = 3100 nM T57392 C32HNI 71541192 IC50 = 6600 nM T57392 C9C0JU 71541193 IC50 = 5600 nM T57392 CD1T5J 71541195 IC50 = 6400 nM T57392 CQ81HF 71541289 IC50 = 7800 nM T57392 CU53JE 71541292 IC50 > 20000 nM T57392 C3RQP5 71542927 IC50 > 10000 nM T57392 C1GUX2 71542931 IC50 > 10000 nM T57392 C0IK7U 71544354 IC50 > 12.5 nM T57392 C83YJF 71544946 IC50 > 50000 nM T57392 CCN01X 71547862 IC50 > 10000 nM T57392 CKB12X 71549359 IC50 > 100000 nM T57392 C4LZM6 71549637 IC50 = 42000 nM T57392 C6JOB5 71549767 IC50 > 100000 nM T57392 CV47CJ 71549769 IC50 = 39000 nM T57392 C5IV9D 71549913 IC50 = 86000 nM T57392 CSHT69 71550657 IC50 > 19000 nM T57392 C9P5KT 71556166 IC50 > 50000 nM T57392 C8JOU5 71556223 IC50 > 50000 nM T57392 C25XGY 71556353 IC50 > 50000 nM T57392 CP0J5L 71556425 IC50 = 33000 nM T57392 CB5QR3 71556493 IC50 = 42000 nM T57392 CIXL34 71556883 IC50 = 38000 nM T57392 CZ3A7E 71556887 IC50 > 50000 nM T57392 CY59CA 71557630 IC50 = 260 nM T57392 CTI52S 71557789 IC50 = 270 nM T57392 CMKH30 71558122 IC50 > 10000 nM T57392 CS8M1O 71558621 IC50 > 10000 nM T57392 CJXK67 71559365 IC50 > 9000 nM T57392 C30ZKJ 71561420 IC50 > 10000 nM T57392 C3L9HK 71562375 IC50 = 251.19 nM T57392 CH49FE 71562477 IC50 = 794.33 nM T57392 CI3KA2 71562588 IC50 = 630.96 nM T57392 C0NIA6 71562591 IC50 = 501.19 nM T57392 CRCT65 71562592 IC50 = 316.23 nM T57392 CFQP86 71562712 IC50 = 5011.87 nM T57392 CS59VG 71562715 IC50 = 1995.26 nM T57392 CE7X9R 71562716 IC50 = 1258.93 nM T57392 CP20LV 71562717 IC50 = 1000 nM T57392 CSYR25 71562833 IC50 = 3981.07 nM T57392 C1Q4JZ 71562837 IC50 = 3981.07 nM T57392 CR8UF1 71563084 IC50 = 840 nM T57392 CLR92N 71579539 IC50 > 100000 nM T57392 C84GAB 71580631 IC50 > 100000 nM T57392 C4S1TN 71580827 IC50 = 50500 nM T57392 C6CHY1 71580912 IC50 = 62100 nM T57392 CUJT21 71582799 IC50 > 10000 nM T57392 CWD2Z5 71585566 IC50 > 10000 nM T57392 CCE7T2 71585568 IC50 > 10000 nM T57392 C4GNJ3 71598545 IC50 > 10000 nM T57392 C1M7JD 71599971 IC50 > 40000 nM T57392 C0WAH3 71602807 IC50 > 30000 nM T57392 C9J0EH 71603917 IC50 > 50000 nM T57392 C8SGK6 71624246 IC50 > 20000 nM T57392 C2WJX0 71626755 IC50 > 50000 nM T57392 C26TXG 71626895 IC50 > 50000 nM T57392 C4DHC9 71626896 IC50 > 50000 nM T57392 CJV92N 71626898 IC50 = 16000 nM T57392 C3XV8I 71626968 IC50 = 33000 nM T57392 CX0VE7 71626971 IC50 > 50000 nM T57392 CDL35U 71655748 IC50 > 5000 nM T57392 CAN6X5 71656574 IC50 = 11000 nM T57392 C61RYH 71659356 IC50 > 30000 nM T57392 CVDB58 71659357 IC50 > 30000 nM T57392 C28EIT 71659358 IC50 > 30000 nM T57392 C8DF4B 71659489 IC50 > 30000 nM T57392 C7Y0RM 71659490 IC50 > 30000 nM T57392 CKR47S 71659491 IC50 > 30000 nM T57392 CAQ2V1 71659492 IC50 > 30000 nM T57392 CJX32Y 71659493 IC50 > 30000 nM T57392 C05JLG 71659494 IC50 > 30000 nM T57392 COS6Q5 71659610 IC50 > 30000 nM T57392 CNVI07 71659611 IC50 > 30000 nM T57392 CUF06Z 71659612 IC50 > 30000 nM T57392 CT9KZ0 71659613 IC50 > 30000 nM T57392 CZFU74 71659614 IC50 > 30000 nM T57392 CC3L1Y 71659615 IC50 > 30000 nM T57392 CF1HA9 71659751 IC50 > 30000 nM T57392 CF8DV2 71659752 IC50 > 30000 nM T57392 CMA4N0 71659753 IC50 > 30000 nM T57392 CFBA41 71659754 IC50 = 1600 nM T57392 CR58TZ 71659755 IC50 > 30000 nM T57392 CVE91N 71659756 IC50 > 30000 nM T57392 CH4VF0 71659894 IC50 > 30000 nM T57392 C53AOG 71659895 IC50 > 30000 nM T57392 C9WC2J 71659896 IC50 > 30000 nM T57392 CTBX46 71659897 IC50 > 30000 nM T57392 CW0Y5N 71659898 IC50 > 30000 nM T57392 CZD71P 71680760 IC50 = 12400 nM T57392 CCXO28 71681727 IC50 = 2600 nM T57392 C23QGT 71681728 IC50 = 4300 nM T57392 CU20IN 71681888 IC50 = 25000 nM T57392 CC7MT2 71681890 IC50 > 30000 nM T57392 CY8VM4 71695585 IC50 > 10000 nM T57392 C8LE5D 71695973 IC50 > 10000 nM T57392 C9I3GO 71714121 IC50 > 50000 nM T57392 CWB3V1 71718136 IC50 = 9400 nM T57392 C0O4ID 71718185 IC50 = 18000 nM T57392 CO7B8C 71720776 IC50 = 4500 nM T57392 CQEH46 71720911 IC50 > 10000 nM T57392 C30NBJ 71722055 IC50 > 10000 nM T57392 CIN10C 71727133 IC50 > 10000 nM T57392 CB53IQ 71727461 IC50 > 10000 nM T57392 CLE15B 71727801 IC50 > 10000 nM T57392 C6USH8 71727930 IC50 > 10000 nM T57392 C1W4DX 71727932 IC50 > 10000 nM T57392 CJZR51 71728054 IC50 > 10000 nM T57392 CQ21ZD 71733911 IC50 > 50000 nM T57392 C56MYK 71739468 IC50 > 30000 nM T57392 CH45ZR 71744719 IC50 > 20000 nM T57392 C60BIX 71763463 IC50 > 10000 nM T57392 C7NKG8 71766070 IC50 = 2500 nM T57392 C5CDM4 71766212 IC50 > 20000 nM T57392 C6P9HZ 71766360 IC50 > 20000 nM T57392 CJHI28 71770158 IC50 = 2310 nM T57392 C9LU5Q 71770282 IC50 = 3460 nM T57392 CTSK68 71811225 IC50 > 10000 nM T57392 CVL54T 71811261 IC50 > 10000 nM T57392 CH8M5Y 71811363 IC50 > 50000 nM T57392 C1WT8V 71811365 IC50 > 50000 nM T57392 COVS02 71812189 IC50 = 150 nM T57392 C5JV1P 71812623 IC50 > 100000 nM T57392 CJH9K3 71814859 IC50 > 10000 nM T57392 CD28XR 71816087 IC50 > 10000 nM T57392 CC4SU1 71817351 IC50 > 10000 nM T57392 CY04LE 71817500 IC50 > 10000 nM T57392 C6EC3O 72163432 IC50 = 24300 nM T57392 CNF81W 72163837 IC50 > 30000 nM T57392 CB2NP7 72165228 IC50 > 20000 nM T57392 C2OV4Z 72189207 IC50 > 10000 nM T57392 CW4E9O 72189514 IC50 = 400 nM T57392 CAVB46 72189515 IC50 = 5000 nM T57392 C4KUM3 72189516 IC50 = 4800 nM T57392 CR5Y6U 72189517 IC50 > 10000 nM T57392 C46FSX 72189518 IC50 > 10000 nM T57392 CBW0G9 72189519 IC50 > 10000 nM T57392 CC0DB5 72189807 IC50 > 10000 nM T57392 CUQ69N 72189808 IC50 > 10000 nM T57392 C1V7PU 72189809 IC50 > 10000 nM T57392 CC1SR3 72189810 IC50 > 10000 nM T57392 C9NCE7 72189811 IC50 > 10000 nM T57392 C2ZF9X 72190130 IC50 > 10000 nM T57392 CXH2S6 72190131 IC50 > 10000 nM T57392 C12KEZ 72190132 IC50 > 10000 nM T57392 CW64OR 72190133 IC50 > 10000 nM T57392 CWT7K2 72205601 IC50 = 4000 nM T57392 CTKQ98 72375000 IC50 > 30000 nM T57392 CL15CY 72375001 IC50 > 30000 nM T57392 CM92XP 72375119 IC50 > 30000 nM T57392 CE46KA 72375120 IC50 > 30000 nM T57392 CHVL93 72375121 IC50 > 30000 nM T57392 CDEN65 72543942 IC50 > 27000 nM T57392 CR9F6I 72543943 IC50 = 2600 nM T57392 CK7DE4 72545105 IC50 > 20000 nM T57392 CA7Y1S 72547022 IC50 > 27000 nM T57392 CW24CT 72547023 IC50 = 15100 nM T57392 C2NCW7 72547024 IC50 > 27000 nM T57392 C7W9JZ 72547025 IC50 = 11800 nM T57392 C1I6VN 72547026 IC50 = 100 nM T57392 CU80HY 72547065 IC50 = 330 nM T57392 CE3X8Y 72547066 IC50 = 5500 nM T57392 CCVG84 72547070 IC50 = 30000 nM T57392 C0Y6IK 72547282 IC50 > 27000 nM T57392 CK50CR 72547283 IC50 = 200 nM T57392 CZI51W 72547284 IC50 > 27000 nM T57392 C3PTC5 72547285 IC50 = 7200 nM T57392 CY5DQ1 72547286 IC50 = 9800 nM T57392 C5XCD4 72547287 IC50 = 2000 nM T57392 CX70JT 72547320 IC50 = 13900 nM T57392 CPSB14 72547529 IC50 = 1900 nM T57392 CY91WF 72547530 IC50 = 700 nM T57392 C48CJQ 72547531 IC50 = 700 nM T57392 CGTC61 72547532 IC50 = 1800 nM T57392 C81YEF 72547533 IC50 > 27000 nM T57392 C4G2UR 72695027 IC50 > 10000 nM T57392 CDFO42 72695136 IC50 > 10000 nM T57392 CK7F6U 72700776 IC50 > 10000 nM T57392 CM75FY 72703989 IC50 > 25000 nM T57392 CPQ34Z 72703991 IC50 = 6100 nM T57392 CBE48L 72707143 IC50 > 10000 nM T57392 C9OQ2I 72710839 IC50 = 12500 nM T57392 C7A5EW 72714054 IC50 > 50000 nM T57392 C7SZ3V 72714058 IC50 > 50000 nM T57392 CI9B8V 72725478 IC50 = 26700 nM T57392 C3J0ZB 72725671 IC50 = 9880 nM T57392 C8QEJ3 72725792 IC50 > 50000 nM T57392 CGM10E 72737641 IC50 > 25000 nM T57392 C7AO4X 72792633 IC50 > 50000 nM T57392 CLK7O4 72792692 IC50 > 50000 nM T57392 C6R8DI 72943374 IC50 > 20000 nM T57392 C59QLH 72943630 IC50 > 20000 nM T57392 CFG97I 72950095 IC50 > 10000 nM T57392 C9WU2M 72950813 IC50 > 100000 nM T57392 C1QMY5 73053248 IC50 > 10000 nM T57392 CH1JK9 73213123 IC50 > 40000 nM T57392 CV6ZT3 73297271 IC50 > 27000 nM T57392 CLA35R 73332001 IC50 = 27000 nM T57392 C7B2VH 73332466 IC50 > 10000 nM T57392 C57LGA 73349098 IC50 > 10000 nM T57392 C80BSO 73352560 IC50 > 20000 nM T57392 CG7R3F 73353420 IC50 > 30000 nM T57392 CM0W7S 73354069 IC50 > 20000 nM T57392 C9WY3B 73386689 Ki = 423 nM T57392 CRA5H6 73389570 IC50 > 10000 nM T57392 C2PAK9 73438493 IC50 > 30000 nM T57392 CDX9R1 73603344 IC50 > 50000 nM T57392 CTMF86 73603391 IC50 > 50000 nM T57392 C7LER5 73669500 IC50 > 50000 nM T57392 CJKB83 73670174 IC50 > 50000 nM T57392 CHV3W1 73774630 IC50 > 30000 nM T57392 CYV4Z6 73890929 IC50 > 100000 nM T57392 CCFI76 73890932 IC50 > 10000 nM T57392 C15QVF 74221424 IC50 > 100000 nM T57392 CZ3TB5 74221949 IC50 > 50000 nM T57392 CW9N8T 74222036 IC50 > 50000 nM T57392 CI58HT 74222429 IC50 = 10000 nM T57392 CUF63H 74223858 IC50 = 17000 nM T57392 C7RAQ4 74538704 IC50 > 20000 nM T57392 CPS18J 75276948 EC50 > 40000 nM T57392 C2G8VR 75593287 IC50 = 11200 nM T57392 CD4IX1 75593344 IC50 = 1400 nM T57392 CB4V1R 76071142 IC50 > 20000 nM T57392 CBAT06 76071144 IC50 > 30000 nM T57392 C7SH1T 76071506 IC50 > 20000 nM T57392 CS87EI 76071624 IC50 > 20000 nM T57392 C9E0PX 76071764 IC50 > 10000 nM T57392 C1Y7HC 76072411 IC50 > 10000 nM T57392 C20YHA 76283431 IC50 > 30000 nM T57392 CHV72I 76283681 IC50 > 20000 nM T57392 CT59ZA 76283684 IC50 > 20000 nM T57392 CE2NP9 76284760 IC50 > 20000 nM T57392 CM9B0T 76309741 IC50 = 23500 nM T57392 C7ZM6V 76310313 IC50 > 39000 nM T57392 C7JAY2 76310561 IC50 = 1100 nM T57392 CQY40K 76310562 IC50 = 2300 nM T57392 CA70YQ 76310589 IC50 > 30000 nM T57392 CY0HD7 76311092 IC50 > 10000 nM T57392 CAT65E 76311096 IC50 = 7600 nM T57392 CF07EK 76313382 IC50 = 12000 nM T57392 C1UOY7 76313414 IC50 = 2900 nM T57392 C8RM5L 76313428 IC50 = 1600 nM T57392 CXC2S5 76313429 IC50 = 8200 nM T57392 CTN57W 76313430 IC50 = 26700 nM T57392 CQFG10 76314530 IC50 > 50000 nM T57392 CX3LZ0 76314702 IC50 = 3200 nM T57392 CJO15N 76316894 IC50 = 18000 nM T57392 C6FX7K 76316938 IC50 = 6500 nM T57392 CT37MX 76316939 IC50 = 3000 nM T57392 C3OP2B 76319044 IC50 > 10000 nM T57392 C6YW3I 76320668 IC50 = 2400 nM T57392 C4G0CX 76320669 IC50 = 18300 nM T57392 CEK3O5 76321713 IC50 > 30000 nM T57392 CNY2D6 76321910 EC50 > 40000 nM T57392 C7Y5QF 76321979 IC50 > 10000 nM T57392 CR05PL 76322043 IC50 = 78800 nM T57392 CQ3CW1 76322044 IC50 > 100000 nM T57392 CYXU43 76322162 IC50 > 30000 nM T57392 CYMO73 76324312 IC50 = 7100 nM T57392 CC8JI7 76324313 IC50 = 4000 nM T57392 CR7FP8 76324529 IC50 = 350 nM T57392 C2SM8Y 76325108 IC50 > 30000 nM T57392 C1HJQ9 76325597 IC50 > 10000 nM T57392 CEAQ91 76327878 IC50 = 6800 nM T57392 CGO16S 76327879 IC50 = 2900 nM T57392 CZE1O7 76327880 IC50 = 7300 nM T57392 CJ9N0S 76328675 IC50 > 30000 nM T57392 C5UMK8 76328829 IC50 > 30000 nM T57392 C8CQ9Y 76328873 IC50 > 30000 nM T57392 CZ9Q2S 76329164 IC50 > 10000 nM T57392 C7Q8YI 76331527 IC50 = 580 nM T57392 CWD5R4 76331595 IC50 = 20000 nM T57392 CZ2CQ7 76332826 IC50 > 10000 nM T57392 C76UKL 76333454 IC50 = 16000 nM T57392 C9QYB2 76335964 IC50 = 400 nM T57392 CE4YP9 76335969 IC50 > 10000 nM T57392 CGE5S3 76336366 EC50 > 40000 nM T57392 CGJM01 76336447 IC50 > 10000 nM T57392 C92WBQ 76336500 IC50 = 18300 nM T57392 CAT95V 76685067 IC50 > 200000 nM T57392 CQT14W 76955651 IC50 = 30000 nM T57392 CWG4T2 78209992 IC50 > 50 nM T57392 CLB1A4 78319901 IC50 > 50000 nM T57392 C86QLE 81689770 IC50 = 4300 nM T57392 C9GQS2 81689815 IC50 > 100000 nM T57392 C3H5XR 82639722 IC50 = 8000 nM T57392 CQMB31 85470872 IC50 > 10000 nM T57392 C15BSO 86270136 IC50 > 10000 nM T57392 CA1CE3 86270720 IC50 > 10000 nM T57392 C9TE7X 86271008 IC50 > 10000 nM T57392 CMZV56 86271009 IC50 > 10000 nM T57392 CXN93A 86271108 IC50 > 10000 nM T57392 C2KHM0 86271111 IC50 > 10000 nM T57392 CZL23E 86271138 IC50 > 30000 nM T57392 C5IR2K 86271238 IC50 > 30000 nM T57392 CN9MO7 86271494 IC50 > 10000 nM T57392 C4T3IW 86272102 IC50 > 100000 nM T57392 C13AJC 86274362 IC50 > 100000 nM T57392 C3OLB1 86274489 IC50 = 88000 nM T57392 CAB78T 86274732 IC50 > 100000 nM T57392 CCU13T 86275207 IC50 > 100000 nM T57392 CJ68CO 86275449 IC50 > 100000 nM T57392 CF4QX9 86278359 IC50 > 10000 nM T57392 CXF9Q3 86279146 IC50 = 28000 nM T57392 C4Y3VP 86279147 IC50 = 20000 nM T57392 CH3FN8 86288905 IC50 > 30000 nM T57392 CKQ71X 86288935 IC50 = 21430 nM T57392 CMKO61 86303027 IC50 = 8000 nM T57392 C3Y9KN 86303187 IC50 = 1900 nM T57392 C6A1DG 86304283 IC50 > 100000 nM T57392 C0IZU4 86304284 IC50 > 100000 nM T57392 C5JFM1 86304285 IC50 > 100000 nM T57392 CKJI10 86304439 IC50 > 100000 nM T57392 CGK31H 86304440 IC50 > 100000 nM T57392 CJ7SI6 86304441 IC50 > 100000 nM T57392 C9EMQ0 86304601 IC50 > 34000 nM T57392 CV4Q5D 86304762 IC50 > 100000 nM T57392 CB5F1W 86343364 IC50 = 14200 nM T57392 CKG7N2 86343365 IC50 = 26400 nM T57392 C9IVM5 86343366 IC50 = 19800 nM T57392 CMXZ65 86346192 IC50 > 10000 nM T57392 CMG39E 86673884 IC50 > 20000 nM T57392 CVJ8L5 86728666 IC50 = 8400 nM T57392 C7OIC6 86762648 IC50 = 9100 nM T57392 CQ45XR 86763358 IC50 > 15848.93 nM T57392 C2U0BG 87055263 IC50 > 10000 nM T57392 CSRU90 87550393 IC50 > 20000 nM T57392 CF67AV 88875879 IC50 > 100000 nM T57392 C8Y9RW 89462922 IC50 > 12.5 nM T57392 C0DRH8 89463724 IC50 > 10 nM T57392 C8SK1N 89463725 IC50 > 12.5 nM T57392 CL30TR 89471870 IC50 > 25000 nM T57392 CA49UY 89726151 IC50 > 30000 nM T57392 CY6K5P 89738540 IC50 > 30000 nM T57392 CIXB02 89738547 IC50 > 30000 nM T57392 CG9CM0 89750383 IC50 = 3100 nM T57392 C2BM9L 89768534 IC50 = 20800 nM T57392 CB4Y7R 89768546 IC50 = 23900 nM T57392 C5MR9K 89777151 IC50 = 19000 nM T57392 CRZ34V 89777258 IC50 = 1300 nM T57392 CZ58KT 89777437 IC50 > 30000 nM T57392 C5S4PX 89777463 IC50 > 30000 nM T57392 CI57QV 89782019 IC50 > 50000 nM T57392 C9I6NQ 89789762 IC50 = 47000 nM T57392 CUS70D 89793496 IC50 > 10000 nM T57392 CP7MZ2 89793516 IC50 > 10000 nM T57392 C9X5OT 89793519 IC50 > 10000 nM T57392 C96EWN 89795484 IC50 > 10000 nM T57392 CWO58S 89795501 IC50 > 10000 nM T57392 CIQ53M 89795553 IC50 > 10000 nM T57392 C5GQL0 89795796 IC50 > 10000 nM T57392 CGD0S5 89825760 IC50 > 20000 nM T57392 CA34IP 89826402 IC50 > 185000 nM T57392 C7GC8K 89826796 IC50 > 20000 nM T57392 C1IA0Q 89826982 IC50 > 20000 nM T57392 CMJY71 89827041 IC50 > 20000 nM T57392 C16AXO 89846366 IC50 > 50000 nM T57392 CEK2I7 89846957 IC50 > 20000 nM T57392 C4MJ6O 89846958 IC50 > 50000 nM T57392 CMS6X4 89931025 IC50 > 20000 nM T57392 CQ5HZ7 89996234 IC50 > 50000 nM T57392 CI54WQ 89996408 IC50 > 10000 nM T57392 CJ65EF 90012001 IC50 > 10000 nM T57392 COVK20 90142631 IC50 > 40000 nM T57392 CY5IC7 90252834 IC50 = 2800 nM T57392 C84NVA 90252850 IC50 > 50000 nM T57392 CBY46O 90252851 IC50 > 50000 nM T57392 CNVA50 90252852 IC50 > 50000 nM T57392 CRN8G1 90253396 IC50 > 20000 nM T57392 CE4IT5 90408860 IC50 > 10000 nM T57392 CB0RP3 90410604 IC50 > 10000 nM T57392 CQ8ZW3 90410911 IC50 > 10000 nM T57392 CD5W6K 90417914 IC50 = 65000 nM T57392 CJE7P5 90467013 IC50 > 50000 nM T57392 CX6DQ4 90467014 IC50 > 50000 nM T57392 C7D2UK 90467156 IC50 > 50000 nM T57392 CV75ZC 90467159 IC50 > 50000 nM T57392 C3RO1M 90467162 IC50 > 50000 nM T57392 CF30KA 90643570 IC50 > 100000 nM T57392 CGS36U 90644505 IC50 > 25000 nM T57392 CYE3G5 90644506 IC50 = 17100 nM T57392 CDE57X 90644507 IC50 > 25000 nM T57392 CV53YI 90644508 IC50 > 10000 nM T57392 C1S8PM 90644647 IC50 > 30000 nM T57392 C5WDB0 90644648 IC50 > 30000 nM T57392 C5O8HN 90644762 IC50 = 26300 nM T57392 CY4PB3 90644766 IC50 > 30000 nM T57392 CL5UB3 90644769 IC50 = 28300 nM T57392 C6AMK9 90644770 IC50 = 12500 nM T57392 CAVN86 90644773 IC50 = 27900 nM T57392 CEZK64 90645309 IC50 > 20000 nM T57392 CXUH46 90645310 IC50 > 20000 nM T57392 C0NM1C 90645311 IC50 = 1900 nM T57392 CL0O7Q 90645312 IC50 > 20000 nM T57392 CHP74S 90654587 IC50 > 10000 nM T57392 C96YCU 90654600 IC50 > 25000 nM T57392 CIL2W9 90664452 IC50 = 4800 nM T57392 CSDO81 90664458 IC50 > 10000 nM T57392 CQT69X 90664721 IC50 > 100000 nM T57392 CN3A1P 90664848 IC50 = 20500 nM T57392 CJ01LW 90664969 IC50 = 12200 nM T57392 C01UNB 90665166 IC50 > 10000 nM T57392 CG98QO 90665194 IC50 = 5400 nM T57392 C02PLA 90665208 IC50 > 100000 nM T57392 CXEJ32 90665986 IC50 > 30000 nM T57392 CDQ56W 90665987 IC50 > 30000 nM T57392 C5E2FJ 90665988 IC50 > 30000 nM T57392 CXEK45 90681222 IC50 > 30000 nM T57392 C8H4KE 90681223 IC50 > 30000 nM T57392 CA9PL8 91663316 IC50 > 30000 nM T57392 C65ANP 91666625 IC50 > 40000 nM T57392 C26BZK 91666633 IC50 > 10000 nM T57392 C9ETC1 91666645 IC50 = 3100 nM T57392 CUI10E 91666686 IC50 = 30000 nM T57392 C2H7XV 91668260 IC50 > 5000 nM T57392 C4YP6M 91754658 IC50 > 100000 nM T57392 C5CKD3 91754690 IC50 > 20000 nM T57392 CZJ6S7 91757962 IC50 = 370 nM T57392 CM95VC 91758806 IC50 = 20000 nM T57392 C5T0FH 91799687 IC50 > 10000 nM T57392 CUX4B6 91809187 IC50 > 60000 nM T57392 CUQ1W0 91810395 IC50 > 50000 nM T57392 CK6E0W 91810397 IC50 = 8400 nM T57392 CWTO83 91810751 IC50 > 10000 nM T57392 CC9B6T 91820646 IC50 > 18000 nM T57392 C3L6KU 91820689 IC50 > 25000 nM T57392 CL7S4U 91844670 IC50 > 10000 nM T57392 C1JPD6 91844700 IC50 > 10000 nM T57392 CSK6Z1 91844707 IC50 = 9800 nM T57392 CH4L7O 91885483 IC50 > 30000 nM T57392 CBG6E7 91885506 IC50 > 5600 nM T57392 C60HAJ 91885643 IC50 = 8200 nM T57392 CU1G3S 91933941 IC50 > 10000 nM T57392 C1SAH3 91971253 IC50 = 58600 nM T57392 CWZX73 91971958 IC50 = 3300 nM T57392 C57QJY 92045044 EC50 > 100000 nM T57392 C38ZID 92045057 IC50 = 5100 nM T57392 CM6VG1 92239323 IC50 > 20000 nM T57392 CY2UI5 101891769 IC50 = 3890 nM T57392 CGB54P 101902999 IC50 = 10000 nM T57392 CG62HP 101903000 IC50 = 5000 nM T57392 C87GEW 102435977 IC50 = 20000 nM T57392 CQ9PN8 102593934 IC50 > 30000 nM T57392 C4Z1OU 110451319 IC50 = 10000 nM T57392 CN57AX 110451673 IC50 > 25000 nM T57392 CYX7T2 117072549 IC50 = 49000 nM T57392 C8F6VO 117604931 IC50 > 100000 nM T57392 CNFW42 117608566 IC50 > 10000 nM T57392 CGL3R6 117614609 IC50 > 100000 nM T57392 CL5OI9 117668598 IC50 > 20000 nM T57392 C5IO0K 117671078 IC50 = 3300 nM T57392 CE8SK5 117671214 IC50 > 20000 nM T57392 CS72RV 117885758 IC50 > 50000 nM T57392 C6Z3NJ 117885766 IC50 > 50000 nM T57392 CKU6S4 117885912 IC50 > 50000 nM T57392 C89EQN 117897570 IC50 > 7200 nM T57392 C9KV7L 117993993 IC50 > 50000 nM T57392 CNV24M 117993998 IC50 > 50000 nM T57392 CGBO72 118016229 IC50 > 20000 nM T57392 C3TBD8 118103460 IC50 > 30000 nM T57392 CZR2Q1 118103881 IC50 = 24800 nM T57392 CL15XC 118103886 IC50 > 30000 nM T57392 CI9Q2H 118103892 IC50 > 30000 nM T57392 CI3KM2 118103909 IC50 > 30000 nM T57392 CAIU03 118104096 IC50 > 30000 nM T57392 CIL65X 118104099 IC50 > 30000 nM T57392 CTA7N8 118107436 IC50 = 1260 nM T57392 CMX3U8 118107483 IC50 >= 5000 nM T57392 CWR6I1 118112300 IC50 = 32000 nM T57392 CNM1W9 118141977 IC50 > 50000 nM T57392 C56INY 118142016 IC50 > 50000 nM T57392 CN1LC9 118142017 IC50 > 50000 nM T57392 CZ0E5W 118142030 IC50 > 10000 nM T57392 CW5N0O 118142047 IC50 > 100000 nM T57392 CWL5J8 118174040 IC50 > 30000 nM T57392 CS6Y1X 118174075 IC50 > 30000 nM T57392 CF38UC 118174137 IC50 > 20000 nM T57392 CKXC27 118174156 IC50 > 20000 nM T57392 CDA16S 118174232 IC50 = 8500 nM T57392 CS7ER1 118174312 IC50 > 30000 nM T57392 CR4DE7 118175009 IC50 > 10000 nM T57392 C2U3TJ 118208018 IC50 > 20000 nM T57392 C6HSC3 118217854 IC50 > 10000 nM T57392 CEKH57 118217858 IC50 > 10000 nM T57392 CRM37Z 118223719 IC50 > 25000 nM T57392 CEN18L 118224069 IC50 = 16700 nM T57392 CT42ZR 118261815 IC50 > 50000 nM T57392 C3R9TY 118324047 IC50 > 10000 nM T57392 C7AO1M 118324066 IC50 > 10000 nM T57392 CPO08K 118344339 IC50 > 20000 nM T57392 CTCQ02 118344344 IC50 > 20000 nM T57392 C1HX3A 118344346 IC50 > 20000 nM T57392 CI7P6J 118344348 IC50 > 20000 nM T57392 C8J1PY 118344351 IC50 > 20000 nM T57392 CAWZ16 118344383 IC50 > 20000 nM T57392 CSUK24 118344385 IC50 > 20000 nM T57392 CA1YM6 118344504 IC50 > 20000 nM T57392 CC3N6Z 118344616 IC50 > 20000 nM T57392 CC0RD7 118345442 IC50 > 20000 nM T57392 CK43EA 118345549 IC50 > 20000 nM T57392 C0MCW3 118346170 IC50 > 20000 nM T57392 CRZ5N1 118368912 IC50 > 50000 nM T57392 CBIR89 118389918 IC50 = 14200 nM T57392 CC7R5L 118399605 IC50 > 20000 nM T57392 CMK5Y8 118399612 IC50 < 1000 nM T57392 CN7EP4 118399635 IC50 < 1000 nM T57392 CG4KD8 118399643 IC50 < 1000 nM T57392 C4WAQ6 118399787 IC50 = 12000 nM T57392 CL6IV1 118440826 IC50 = 5100 nM T57392 CAXT13 118441135 IC50 < 1000 nM T57392 CHIL17 118441142 IC50 = 3500 nM T57392 CR7DJ0 118453722 IC50 > 50000 nM T57392 CK1Z7I 118462026 IC50 > 50000 nM T57392 CM2NH5 118478848 IC50 > 30000 nM T57392 CRV8S3 118478927 IC50 > 10000 nM T57392 CL32JE 118478933 IC50 > 10000 nM T57392 C5S1HZ 118478972 IC50 > 10000 nM T57392 C8G9HP 118478986 IC50 > 10000 nM T57392 CBV89G 118478994 IC50 > 10000 nM T57392 CK0ER5 118478999 IC50 > 10000 nM T57392 CU25KC 118479000 IC50 > 10000 nM T57392 CW07IS 118479006 IC50 > 10000 nM T57392 C3ZAV0 118479034 IC50 > 10000 nM T57392 C4W6ZS 118479038 IC50 > 10000 nM T57392 CRG24C 118479053 IC50 > 10000 nM T57392 CD4ME1 118479123 IC50 > 10000 nM T57392 CB0XM2 118479161 IC50 > 10000 nM T57392 C18NTQ 118479199 IC50 > 10000 nM T57392 CJ0Z1Y 118479222 IC50 > 10000 nM T57392 CP0U6Y 118479229 IC50 > 10000 nM T57392 C3A6HD 118479231 IC50 > 10000 nM T57392 CJ14CR 118479241 IC50 > 10000 nM T57392 C1FO3N 118479293 IC50 > 10000 nM T57392 CF02TZ 118479295 IC50 > 10000 nM T57392 C90TED 118479305 IC50 > 10000 nM T57392 C7I9RC 118479316 IC50 > 10000 nM T57392 CRC4F6 118479354 IC50 > 10000 nM T57392 CRCV51 118479359 IC50 > 10000 nM T57392 CJL5W0 118479428 IC50 > 10000 nM T57392 CS2VA7 118479440 IC50 > 10000 nM T57392 CJ9P0M 118479445 IC50 > 10000 nM T57392 C3U1RB 118479452 IC50 > 10000 nM T57392 CBJ28X 118483320 Ki = 720 nM T57392 C8PU5O 118491249 IC50 > 10000 nM T57392 C3KAO6 118491258 IC50 = 16000 nM T57392 CINA28 118492166 IC50 = 12000 nM T57392 CJ9Z0S 118496546 IC50 > 50000 nM T57392 C7AYV5 118540795 IC50 = 8830 nM T57392 CB41MH 118560618 IC50 = 15000 nM T57392 C78LNX 118572065 IC50 > 30000 nM T57392 C0XJT5 118626089 IC50 > 100000 nM T57392 CRS34C 118705500 IC50 > 100000 nM T57392 CVNL09 118706404 IC50 = 15000 nM T57392 CLUN23 118706414 IC50 > 20000 nM T57392 C2BG1F 118706537 IC50 = 530 nM T57392 C2WP6X 118706538 IC50 = 8700 nM T57392 CZE4U0 118706539 IC50 = 4000 nM T57392 CX8I0G 118706540 IC50 = 1000 nM T57392 C2O7GE 118707553 IC50 > 20000 nM T57392 C8S9VW 118707562 IC50 > 20000 nM T57392 CS4R3B 118707826 IC50 > 30000 nM T57392 CR8VJ2 118708873 IC50 > 5000 nM T57392 CL2VY5 118708881 IC50 > 5000 nM T57392 CB5F2O 118708929 IC50 > 5000 nM T57392 C8M3JX 118708934 IC50 > 5000 nM T57392 C9W3LI 118708938 IC50 > 5000 nM T57392 CEAK31 118708939 IC50 > 5000 nM T57392 CMX6S5 118709259 IC50 > 20000 nM T57392 CG19YT 118709623 IC50 = 18000 nM T57392 CT1J7Y 118709777 IC50 = 9620 nM T57392 CD34IY 118710582 IC50 = 11000 nM T57392 CD1O7G 118710583 IC50 = 1000 nM T57392 CT91SV 118711722 IC50 > 20000 nM T57392 C4VAE0 118713757 IC50 = 10 nM T57392 C84GOU 118713773 IC50 = 2100 nM T57392 C2LY9D 118713799 IC50 = 620 nM T57392 CMO2V7 118713801 IC50 = 2340 nM T57392 C9LKI0 118713803 IC50 = 130 nM T57392 C2OZ7H 118713805 IC50 = 20 nM T57392 CM4P8X 118713806 IC50 = 13700 nM T57392 C7EXQ9 118713807 IC50 = 1880 nM T57392 CUM74B 118716060 IC50 > 10000 nM T57392 CLGD29 118720097 IC50 > 10000 nM T57392 C4LW6I 118720885 IC50 > 40000 nM T57392 C9SF2E 118720891 IC50 > 24000 nM T57392 C8VYR0 118721373 IC50 = 370 nM T57392 CFL73Q 118724203 IC50 > 50000 nM T57392 C6RXB2 118729222 IC50 = 18000 nM T57392 C9HFE1 118730345 IC50 > 10000 nM T57392 C6HV3B 118730351 IC50 > 10000 nM T57392 C3LZM9 118730352 IC50 = 7400 nM T57392 C6B4XD 118730937 IC50 = 7100 nM T57392 CO81CK 118730940 IC50 > 20000 nM T57392 C27FIO 118730943 IC50 > 20000 nM T57392 C6OEU2 118733374 IC50 > 50000 nM T57392 C4G3YC 118734875 IC50 > 30000 nM T57392 C9AIE1 118734876 IC50 > 30000 nM T57392 C0SM3L 118735340 IC50 < 5000 nM T57392 CAN90V 118735353 IC50 > 100000 nM T57392 C4XY9I 118735354 IC50 > 100000 nM T57392 C1XL4S 118735355 IC50 = 27000 nM T57392 CB57VC 118737720 IC50 > 50000 nM T57392 C15QMA 118737724 IC50 > 50000 nM T57392 C1MHT0 118737725 IC50 > 50000 nM T57392 C5BOQ1 118753201 Ki > 30000 nM T57392 C87ZPY 118796358 IC50 > 50000 nM T57392 CIPQ86 118861736 EC50 > 100000 nM T57392 CR71BE 118861737 EC50 > 100000 nM T57392 CDSY04 118861738 EC50 = 4940 nM T57392 C9WBY6 118861778 EC50 = 41200 nM T57392 CELZ36 118866105 IC50 = 20000 nM T57392 C14DLY 118872292 Ki = 3130 nM T57392 CM59EQ 118917669 IC50 > 30000 nM T57392 C6J8YF 118917671 IC50 > 30000 nM T57392 C2RBF7 118918048 IC50 = 2000 nM T57392 CC4LA1 118953461 IC50 = 1200 nM T57392 C8L1QI 118959080 IC50 > 5000 nM T57392 C9LR8Z 118965395 IC50 > 100000 nM T57392 C13EIL 118967091 IC50 = 120 nM T57392 CE3CN6 118971057 IC50 < 100 nM T57392 C4K3PR 118987036 IC50 > 25000 nM T57392 COS3K9 121304408 IC50 > 5000 nM T57392 C9G3ZJ 121304414 IC50 > 7000 nM T57392 C4RD9Y 121304424 IC50 = 5700 nM T57392 C1PKR0 121304441 IC50 > 3000 nM T57392 CC3MP6 121304452 IC50 > 3000 nM T57392 CW68KD 121304458 IC50 = 130 nM T57392 CPB58L 121304467 IC50 > 9000 nM T57392 COB2X5 121304477 IC50 > 7000 nM T57392 CZ0BI4 121304484 IC50 > 38000 nM T57392 CW51NQ 121304485 IC50 = 1300 nM T57392 CX1DQ6 121304488 IC50 > 6000 nM T57392 C7NLV2 121304500 IC50 > 10000 nM T57392 CPNV43 121304527 IC50 = 1200 nM T57392 CQ2UM4 121304538 IC50 > 17000 nM T57392 C1AB6P 121304551 IC50 = 700 nM T57392 CN05ZQ 121304574 IC50 > 17000 nM T57392 CU0M7B 121304590 IC50 = 1300 nM T57392 CX5MO3 121304598 IC50 = 2000 nM T57392 C31AEQ 121304649 IC50 = 600 nM T57392 C2VTK5 121304654 IC50 > 10000 nM T57392 C6IB0P 121304685 IC50 > 21000 nM T57392 CXC70Q 121304711 IC50 > 1000 nM T57392 C6C9EF 121304827 IC50 = 450 nM T57392 CU4CW1 121313969 IC50 > 50000 nM T57392 C65ZYO 121332604 IC50 > 3000 nM T57392 C92NOH 121332654 IC50 > 3000 nM T57392 CNBH32 121332727 IC50 > 3000 nM T57392 C9Q2ND 121333973 IC50 > 15000 nM T57392 C6TBD2 121345502 IC50 > 50000 nM T57392 C4CPO3 121398401 IC50 > 25000 nM T57392 C59ORZ 121398668 IC50 > 10000 nM T57392 CV9TX1 121399281 IC50 = 31650 nM T57392 C2WD1Q 121407246 IC50 = 30400 nM T57392 C9CV7H 121411850 IC50 > 20000 nM T57392 CU3BI0 121412063 IC50 > 20000 nM T57392 CQZ9W3 121414283 IC50 > 25000 nM T57392 C91PVZ 121428416 IC50 > 10000 nM T57392 C3KNZ5 121439991 IC50 > 50000 nM T57392 CV5R4G 121470704 IC50 > 50000 nM T57392 C85HZL 121470706 IC50 > 50000 nM T57392 C09QGL 121470709 IC50 > 50000 nM T57392 C3OL2H 121480641 IC50 > 50000 nM T57392 CD89ZC 121480642 IC50 > 50000 nM T57392 CHD26A 121596332 IC50 > 20000 nM T57392 CP52DJ 121596967 IC50 = 12710 nM T57392 C2AWE9 122178128 IC50 = 20 nM T57392 C9WB6E 122179416 IC50 > 100000 nM T57392 CYFA75 122179419 IC50 > 100000 nM T57392 CNGQ19 122179477 IC50 > 10000 nM T57392 C83WUQ 122181896 IC50 < 780 nM T57392 CDU51C 122181897 IC50 < 780 nM T57392 CO31SP 122181898 IC50 < 780 nM T57392 CM8YU5 122181899 IC50 < 780 nM T57392 C0CPA8 122181900 IC50 = 680 nM T57392 CT34BU 122181901 IC50 < 780 nM T57392 CIG56Y 122181903 IC50 < 780 nM T57392 C8M4CH 122182156 IC50 = 2900 nM T57392 CTJO50 122184561 IC50 = 6500 nM T57392 CZ1MA3 122184562 IC50 = 15000 nM T57392 CH37IW 122184563 IC50 = 2400 nM T57392 C5JTD9 122184564 IC50 > 50000 nM T57392 C0I3YT 122184610 IC50 = 68 nM T57392 C3SPQ8 122184611 IC50 = 44 nM T57392 C6AZC1 122184743 IC50 = 1900 nM T57392 CQA8B2 122187067 IC50 > 100000 nM T57392 CS5CF1 122187069 IC50 > 100000 nM T57392 C14FGL 122187534 IC50 > 20000 nM T57392 CB7IJ0 122188138 IC50 > 20000 nM T57392 C9TF8M 122190433 IC50 > 30000 nM T57392 CCD9E8 122190697 IC50 = 5560 nM T57392 CF0KD5 122190700 IC50 = 9640 nM T57392 C8GHY3 122190972 IC50 > 30000 nM T57392 CTI2V5 122192293 IC50 > 40000 nM T57392 C4NUY0 122192382 IC50 > 10000 nM T57392 C1MVP5 122192989 IC50 > 50000 nM T57392 CLHV68 122192990 IC50 > 50000 nM T57392 C1N0HP 122193176 IC50 > 30000 nM T57392 CV8J6N 122193177 IC50 > 30000 nM T57392 CB8MH7 122193179 IC50 > 30000 nM T57392 CQX7P1 122195090 IC50 > 2000 nM T57392 CUE4R9 122195192 IC50 > 20000 nM T57392 CNF81V 122195193 IC50 > 20000 nM T57392 CCP5U2 122195692 IC50 > 30000 nM T57392 CSR2O7 122195839 IC50 = 600 nM T57392 C62JEW 122196028 IC50 > 10000 nM T57392 C53POD 122196029 IC50 > 10000 nM T57392 CCP15H 122197303 IC50 = 4170 nM T57392 C32PNV 122234475 IC50 > 20000 nM T57392 C1C9LI 122246967 IC50 = 6100 nM T57392 CGT12J 122419159 IC50 > 30000 nM T57392 C2F6EH 122456006 IC50 > 30000 nM T57392 C6QHB4 122484585 IC50 > 50000 nM T57392 COX7E3 122510453 IC50 > 20000 nM T57392 CLM7K3 122604539 IC50 > 50000 nM T57392 C01JHI 122604566 IC50 = 35000 nM T57392 CU2K4P 122650372 IC50 > 10000 nM T57392 C3RCU4 122650378 IC50 = 9610 nM T57392 CS47AD 122650581 IC50 > 10000 nM T57392 C85JKN 122668190 IC50 = 16800 nM T57392 CD6X5P 122669265 IC50 > 20000 nM T57392 C86VYP 122670110 IC50 > 30000 nM T57392 C1YK2E 122678192 IC50 > 20000 nM T57392 CK7W8B 123132907 IC50 = 157 nM T57392 CRW0C2 123132915 IC50 = 334 nM T57392 CSLF20 123226629 IC50 > 30000 nM T57392 C7ZJ8U 123295297 IC50 > 30000 nM T57392 CT9K0V 124000588 IC50 > 10000 nM T57392 C6CA4O 124088406 IC50 = 73000 nM T57392 C5ZY7L 124114343 IC50 > 50000 nM T57392 CPO7N5 124125214 IC50 = 4900 nM T57392 C4VT3O 124127413 IC50 = 2000 nM T57392 CZEC76 124147932 IC50 > 50000 nM T57392 CEK31I 124148318 IC50 > 30000 nM T57392 C5H2QB 124150512 IC50 > 50000 nM T57392 C7TOU4 124175991 IC50 > 10000 nM T57392 C53AYP 124176028 IC50 > 10000 nM T57392 CL7K0C 124176200 IC50 > 10000 nM T57392 CYD04K 124176232 IC50 > 10000 nM T57392 CMS9P1 124176233 IC50 > 10000 nM T57392 C7EQH8 124176242 IC50 > 10000 nM T57392 CGJH79 124176281 IC50 > 10000 nM T57392 CCYK63 124176287 IC50 > 10000 nM T57392 CWF7N2 124176288 IC50 > 10000 nM T57392 CK0B3W 124176291 IC50 > 10000 nM T57392 CNC17W 124176295 IC50 > 10000 nM T57392 CMG02Z 124176321 IC50 > 10000 nM T57392 CDS92J 126483508 IC50 > 50000 nM T57392 CP8W0X 126533801 IC50 > 1000 nM T57392 CIV7R0 126533969 IC50 > 17000 nM T57392 CI97TU 126533981 IC50 > 2000 nM T57392 CIAD86 126534204 IC50 > 20000 nM T57392 C4R7XU 126534291 IC50 > 3000 nM T57392 CVBX50 126534373 IC50 > 3000 nM T57392 CFA3D6 126534516 IC50 > 5000 nM T57392 C0WUJ5 126534771 IC50 > 1000 nM T57392 CX9LM7 126534859 IC50 > 15000 nM T57392 C6DLR7 126534986 IC50 > 1000 nM T57392 C9Q0VB 126535075 IC50 > 16000 nM T57392 CIZC84 126535109 IC50 > 25000 nM T57392 CTAG09 126567264 IC50 > 25000 nM T57392 C5QT4N 126567306 IC50 > 25000 nM T57392 C2LAM7 126591927 IC50 > 30000 nM T57392 CZ3TD0 126651203 IC50 > 50000 nM T57392 C0LTB9 126651349 IC50 > 50000 nM T57392 C45OVL 126693206 IC50 = 3400 nM T57392 CS1B2E 127020968 IC50 > 10000 nM T57392 CB2ZK5 127026165 IC50 > 30000 nM T57392 C7J5VX 127026166 IC50 > 30000 nM T57392 C9XU8I 127026167 IC50 > 30000 nM T57392 CU32KG 127026289 IC50 = 16750 nM T57392 CA42BO 127027101 IC50 > 30000 nM T57392 C09CHL 127027102 IC50 > 30000 nM T57392 CCK36V 127029882 IC50 = 7754 nM T57392 CVC84H 127029883 IC50 = 7624 nM T57392 CFY1P0 127029884 IC50 = 4100 nM T57392 CU8Y7N 127030224 IC50 = 16380 nM T57392 CTEA14 127030225 IC50 = 21305 nM T57392 CLDC46 127031152 IC50 > 30000 nM T57392 C60SMC 127031153 IC50 = 29880 nM T57392 C2POU1 127033963 IC50 > 30000 nM T57392 C2JOP5 127034286 IC50 > 30000 nM T57392 CZ61LK 127034966 IC50 = 398.11 nM T57392 CA0SN5 127034967 IC50 = 2511.89 nM T57392 CP0W4Y 127036068 IC50 > 30000 nM T57392 C0V4SJ 127036359 IC50 > 45000 nM T57392 CWDI07 127037076 IC50 = 14000 nM T57392 C8QIK9 127037551 IC50 > 50000 nM T57392 CB41IW 127037818 IC50 = 21900 nM T57392 CZU7Q2 127037819 IC50 = 88500 nM T57392 C5VF7R 127037821 IC50 = 43700 nM T57392 CI6HK4 127038465 IC50 = 3400 nM T57392 C9Y8VL 127038466 IC50 > 100000 nM T57392 CUBG78 127039139 IC50 > 50000 nM T57392 CLN20Q 127039167 IC50 = 7500 nM T57392 C3O7CA 127039374 IC50 = 734300 nM T57392 CA4ZB8 127039509 IC50 = 93500 nM T57392 C20VKF 127039824 IC50 = 90200 nM T57392 C60HOC 127040550 IC50 = 40000 nM T57392 C34BGK 127040715 IC50 > 30000 nM T57392 C0J8HC 127041348 IC50 > 3000 nM T57392 C7PU6F 127041479 IC50 = 48600 nM T57392 CCU4Z1 127041764 IC50 = 1210 nM T57392 CI5TA6 127041772 IC50 = 5240 nM T57392 C6HB0F 127041783 IC50 = 50400 nM T57392 CQ1U5D 127041786 IC50 = 140100 nM T57392 CCJX69 127041842 IC50 = 18000 nM T57392 CS78AZ 127041951 IC50 > 30000 nM T57392 CU9C4S 127041952 IC50 > 6000 nM T57392 C63OPL 127042084 IC50 = 36100 nM T57392 CQCO27 127046038 IC50 = 26500 nM T57392 C34REM 127046317 IC50 > 30000 nM T57392 C9A1TG 127046557 IC50 > 30000 nM T57392 C57ZRE 127046727 IC50 > 50000 nM T57392 CH6W2T 127046982 IC50 = 3300 nM T57392 C7YML2 127047647 IC50 > 30000 nM T57392 CJH46E 127047680 IC50 > 10000 nM T57392 C48NCK 127047993 IC50 = 10300 nM T57392 C84TQV 127048530 IC50 > 20000 nM T57392 CZV7Q0 127049047 IC50 > 10000 nM T57392 CB54VQ 127049048 IC50 > 10000 nM T57392 C9TUQ2 127049049 IC50 > 10000 nM T57392 CJ8SG3 127049204 IC50 < 10000 nM T57392 C2O5LX 127049804 IC50 = 17330 nM T57392 CUVQ34 127050762 IC50 < 1000 nM T57392 CJP90K 127051009 IC50 = 16500 nM T57392 C9V4EG 127051045 IC50 = 59000 nM T57392 C2QX0V 127051283 IC50 > 20000 nM T57392 C7KZJ2 127052145 IC50 = 16900 nM T57392 C38VGB 127052215 IC50 = 12500 nM T57392 CR7O3H 127052463 IC50 > 20000 nM T57392 C4CRE7 127052464 IC50 > 20000 nM T57392 C75EAL 127052638 IC50 = 19000 nM T57392 C2GY5W 127052655 IC50 = 6300 nM T57392 C5OE2H 127053611 IC50 > 20000 nM T57392 CEC17N 129164665 IC50 = 1000 nM T57392 CY4B7Z 129164668 IC50 = 6000 nM T57392 CAT90Y 129164701 IC50 = 2000 nM T57392 CUB58Q 129164743 IC50 = 3000 nM T57392 C81SHO 129178830 IC50 = 500 nM T57392 CJGR20 129240126 IC50 > 30000 nM T57392 CR8HP6 129281194 IC50 > 10000 nM T57392 CE8TV5 129893260 IC50 = 10000 nM T57392 C9NPD3 129909153 IC50 > 25000 nM T57392 C4LR9M 129909326 IC50 > 25000 nM T57392 CD80OM 129909338 IC50 = 15200 nM T57392 CV3UP6 129909861 IC50 > 30000 nM T57392 CK68CA 130453737 IC50 > 30000 nM T57392 CDV84X 131747741 IC50 > 50000 nM T57392 CV06MU 131801402 IC50 > 25000 nM T57392 C4Z5MQ 131839619 IC50 > 30000 nM T57392 CFC05Q 131954513 IC50 > 30000 nM T57392 CN4RF6 132019596 IC50 > 30000 nM T57392 CZ5H2B 132020452 IC50 > 40000 nM T57392 CP8A1Q 132020575 IC50 > 40000 nM T57392 CE9BL3 132046817 IC50 > 30000 nM T57392 CH8DP7 132220479 IC50 > 20000 nM T57392 C5P4XN 132227197 IC50 > 18000 nM T57392 C1R5SZ 132227201 IC50 > 18000 nM T57392 CGDN94 132275066 IC50 > 10000 nM T57392 CACJ46 132489333 IC50 > 25000 nM T57392 C6Z8BD 132510851 IC50 = 700 nM T57392 CN12VW 132550264 IC50 = 7590 nM T57392 CJE34F 132597748 IC50 > 27000 nM T57392 CZC7S8 133081963 IC50 = 2610 nM T57392 C18GQC 134128280 IC50 > 20000 nM T57392 CO1RW6 134132142 IC50 > 50000 nM T57392 CJOQ95 134134229 IC50 > 50000 nM T57392 CES87G 134135247 IC50 = 27000 nM T57392 CC7OQ2 134135307 IC50 > 50000 nM T57392 CE5TV4 134135453 IC50 = 9400 nM T57392 C3P9IJ 134136137 IC50 = 3000 nM T57392 CDRC75 134136284 IC50 = 10200 nM T57392 CK9MG1 134136380 IC50 = 44000 nM T57392 CYI93Q 134136642 IC50 = 640 nM T57392 C2A7CZ 134138904 IC50 = 20950 nM T57392 CU8BV5 134139688 IC50 > 20000 nM T57392 CH3V9Q 134139925 IC50 > 25000 nM T57392 C8MAB7 134142736 IC50 > 30000 nM T57392 CVC1Y4 134142943 IC50 = 5370 nM T57392 CK13YN 134145788 IC50 = 7800 nM T57392 CFG60Q 134148895 IC50 > 10000 nM T57392 CC43OQ 134149366 IC50 > 50000 nM T57392 CA5B2J 134150245 IC50 > 50000 nM T57392 C0S2VH 134150637 IC50 > 17000 nM T57392 C6NYU2 134150754 IC50 > 5000 nM T57392 COPA84 134151189 IC50 = 18000 nM T57392 C9NI7K 134151534 IC50 = 7750 nM T57392 CZH50T 134151855 IC50 = 25650 nM T57392 C8PT9W 134152052 IC50 > 30000 nM T57392 CY54BL 134152502 IC50 = 400 nM T57392 CKU7X4 134152809 IC50 = 8600 nM T57392 CP41RT 134154065 IC50 >= 20000 nM T57392 C0LGI2 134154676 IC50 = 25700 nM T57392 CZV9B3 134154775 IC50 > 30000 nM T57392 CBPN64 134154817 IC50 = 3800 nM T57392 CJ0UG1 134155310 IC50 = 24200 nM T57392 CTX8Q6 134155895 IC50 < 300 nM T57392 CA49BH 134156727 IC50 > 50000 nM T57392 C7H8GQ 134157229 IC50 > 10000 nM T57392 CNS38M 134157776 IC50 = 15750 nM T57392 CK7B0U 134304087 IC50 > 10000 nM T57392 CX62UZ 134304119 IC50 > 10000 nM T57392 CUDY24 134304129 IC50 > 10000 nM T57392 CO5I4B 134304177 IC50 > 10000 nM T57392 CRD52S 134324842 IC50 > 10000 nM T57392 C17NBC 134325016 IC50 > 10000 nM T57392 CVR60G 134539903 IC50 > 25000 nM T57392 C20HAT 134585236 IC50 = 42000 nM T57392 C6W3VL 134585536 IC50 = 23000 nM T57392 CRL3O8 134585831 IC50 = 36000 nM T57392 CZB7I6 134821685 IC50 > 10000 nM T57392 CDC38O 134823958 IC50 = 200 nM T57392 CQI48P 135192983 IC50 > 30000 nM T57392 CT0GQ6 135197577 IC50 > 10000 nM T57392 C87VKA 135197594 IC50 > 10000 nM T57392 CQXS07 135197635 IC50 > 10000 nM T57392 C7KXF1 135197643 IC50 > 10000 nM T57392 CS4BM3 135236903 IC50 > 50000 nM T57392 CNEY95 135285657 IC50 = 5000 nM T57392 CA2OV3 135306913 IC50 > 50000 nM T57392 CH9RX5 135313574 IC50 = 355 nM T57392 CCJ97K 135313618 IC50 = 258 nM T57392 C76OJC 135313705 IC50 > 20000 nM T57392 C2L6PH 135313715 IC50 = 377 nM T57392 CO4W2L 135313730 IC50 = 67800 nM T57392 CQBZ60 135313773 IC50 = 32 nM T57392 C3K2RL 135313899 IC50 = 577 nM T57392 CMR34P 135313919 IC50 > 20000 nM T57392 CR6K4Q 135313963 IC50 = 1450 nM T57392 C9FNU5 135313965 IC50 > 20000 nM T57392 C75MZN 135314048 IC50 = 100000 nM T57392 CL12JU 135314107 IC50 = 100000 nM T57392 CPTO20 135314108 IC50 = 100000 nM T57392 C8Q4JP 135314141 IC50 = 3320 nM T57392 CXN1C7 135314251 IC50 = 709 nM T57392 CBQ01J 135314252 IC50 = 453 nM T57392 C9OZ3G 135314329 IC50 = 660 nM T57392 C46IBJ 135314337 IC50 = 507 nM T57392 CWI13E 135314362 IC50 = 100000 nM T57392 CI73PJ 135314386 IC50 = 84 nM T57392 CM3KV6 135314388 IC50 = 48 nM T57392 CY24QI 135314390 IC50 = 254 nM T57392 CD64BJ 135314469 IC50 = 403 nM T57392 CW3DO8 135315463 IC50 > 50000 nM T57392 C75MTX 135315494 IC50 > 50000 nM T57392 C7K4PA 135412054 IC50 > 20000 nM T57392 C31VAN 135412231 IC50 > 20000 nM T57392 CIS9K5 135421564 IC50 > 10000 nM T57392 C1KUD6 135429838 IC50 = 234000 nM T57392 CZ4GP6 135446244 IC50 > 20000 nM T57392 C3RX6B 135530418 IC50 = 5700 nM T57392 CKF13W 135546072 IC50 > 10000 nM T57392 C8R4FB 135546884 IC50 > 20000 nM T57392 CY4MV6 135566354 IC50 > 50000 nM T57392 C8DX9H 135567148 IC50 > 25000 nM T57392 C23IWG 135567151 IC50 > 25000 nM T57392 CCNH91 135743577 IC50 > 10000 nM T57392 CCK5I3 135883253 IC50 > 10000 nM T57392 C14OBQ 135928469 IC50 > 20000 nM T57392 C01HMT 135932346 IC50 = 20000 nM T57392 C4RL7Q 135985508 IC50 > 10000 nM T57392 C1ZT4N 135988927 IC50 = 10000 nM T57392 C86BZJ 135988997 IC50 = 9000 nM T57392 C4HJ7D 136044076 IC50 > 10000 nM T57392 CT57ZH 136069450 IC50 > 50000 nM T57392 CFT9R3 136069453 IC50 > 50000 nM T57392 CRPQ42 136069494 IC50 > 100000 nM T57392 CK8Z3V 136069521 IC50 > 50000 nM T57392 CPY1B2 136069522 IC50 > 50000 nM T57392 CX0OM4 136069523 IC50 > 50000 nM T57392 C6EU4D 136069524 IC50 > 50000 nM T57392 CQA2Z1 136069531 IC50 > 50000 nM T57392 CCH31A 136069532 IC50 > 50000 nM T57392 CQ1FS4 136069563 IC50 > 50000 nM T57392 C69JHW 136117992 IC50 = 560 nM T57392 CGX6C4 136173253 IC50 > 50000 nM T57392 CC52HL 136189674 IC50 > 20000 nM T57392 CQTB32 136205798 IC50 > 10000 nM T57392 CV8QP3 136205832 IC50 > 50000 nM T57392 CB93EM 136205833 IC50 > 50000 nM T57392 CBS97C 136239447 IC50 = 80 nM T57392 CC8Q2D 136375233 IC50 > 1000 nM T57392 C4OVP2 136416802 IC50 > 50000 nM T57392 C7ZCT8 136416815 IC50 > 50000 nM T57392 C95TJH 136632047 IC50 > 10000 nM T57392 CI94YQ 136982007 IC50 > 10000 nM T57392 CK4CM2 137028369 IC50 > 50000 nM T57392 C7TAZ5 137142885 IC50 > 10000 nM T57392 CO6WA9 137313834 IC50 = 18400 nM T57392 CE1G4P 137333984 IC50 = 1600 nM T57392 C0PL4B 137434175 IC50 > 30000 nM T57392 C8V9ER 137440575 IC50 = 23000 nM T57392 CS34IR 137628304 IC50 > 25000 nM T57392 C9ACX4 137628305 IC50 < 10000 nM T57392 CP2C1J 137628306 IC50 > 25000 nM T57392 CDGB50 137628309 IC50 < 10000 nM T57392 CW8ZR6 137628310 IC50 < 10000 nM T57392 C48QKY 137628311 IC50 < 10000 nM T57392 CH5AV6 137628312 IC50 < 10000 nM T57392 CU9O3A 137628639 IC50 > 20000 nM T57392 CEZT29 137628641 IC50 > 10000 nM T57392 C6B5US 137628648 IC50 > 10000 nM T57392 C3A6PQ 137628670 IC50 > 10000 nM T57392 C6JO4G 137631841 IC50 = 12000 nM T57392 C6MRU3 137633431 IC50 = 434 nM T57392 CV8M3P 137633531 IC50 = 6210 nM T57392 CNU3O7 137634107 IC50 = 629 nM T57392 COD07I 137634464 IC50 = 90 nM T57392 CE9O8V 137634616 IC50 = 12000 nM T57392 CT8E0M 137635041 IC50 = 189 nM T57392 CP07AG 137635043 IC50 = 14000 nM T57392 CYL39G 137635979 IC50 > 10000 nM T57392 CR9IZ6 137637770 IC50 = 400 nM T57392 CDBT63 137637838 IC50 = 141 nM T57392 C21YPG 137638242 IC50 = 217 nM T57392 C2Y9HF 137638913 IC50 = 12000 nM T57392 C8WO2G 137639251 IC50 = 1170 nM T57392 CF5TI6 137639661 IC50 = 6800 nM T57392 CYPQ38 137640446 IC50 = 1750 nM T57392 CV85YQ 137640474 IC50 = 2720 nM T57392 CKL78U 137640727 IC50 = 12590 nM T57392 C0Q4IM 137641652 IC50 = 2610 nM T57392 CYW61U 137641749 IC50 = 510 nM T57392 CH21YK 137642640 IC50 < 200 nM T57392 CR9C5G 137642830 IC50 <= 20000 nM T57392 CO8V4W 137642907 IC50 = 15000 nM T57392 CUB38E 137642944 IC50 = 1000 nM T57392 CJT81N 137643054 IC50 = 13000 nM T57392 CPW7T0 137643121 IC50 = 32100 nM T57392 C58ISN 137643139 IC50 = 3200 nM T57392 C1FU3P 137643308 IC50 = 14000 nM T57392 CVC3S2 137643317 IC50 = 657 nM T57392 C9BF0V 137643369 IC50 = 14000 nM T57392 CI2F1B 137644335 IC50 = 1160 nM T57392 CU91LQ 137644813 IC50 = 2220 nM T57392 CN97GA 137645181 IC50 > 10000 nM T57392 CKT2R4 137646125 IC50 = 354 nM T57392 CU47YW 137646415 IC50 = 16000 nM T57392 C5IHS8 137646440 IC50 = 16000 nM T57392 CN4U1A 137646732 IC50 > 30000 nM T57392 CRA48Q 137647184 IC50 = 494 nM T57392 CLT73G 137647199 IC50 = 13230 nM T57392 CXS2U7 137647336 IC50 = 318 nM T57392 C42DRJ 137647643 IC50 = 348 nM T57392 CLAR76 137647645 IC50 = 853 nM T57392 CGW71J 137647660 IC50 > 50000 nM T57392 CUDM82 137647787 IC50 = 9700 nM T57392 C4AKD7 137647838 IC50 = 345 nM T57392 C5AT7D 137649062 IC50 = 17000 nM T57392 C04JSE 137649716 IC50 = 44500 nM T57392 C8N9CH 137650363 IC50 = 4150 nM T57392 CL7ZX9 137651411 IC50 = 2700 nM T57392 CD9ZN4 137651429 IC50 = 2530 nM T57392 C6GJA5 137651722 IC50 = 45000 nM T57392 C2JBS1 137651899 IC50 > 100000 nM T57392 C2L7ZT 137652982 IC50 = 145 nM T57392 CKV03G 137653074 IC50 > 30000 nM T57392 C38FXZ 137653443 IC50 > 20000 nM T57392 CV59RY 137654290 IC50 = 2040 nM T57392 CMXL93 137655135 IC50 > 10000 nM T57392 CX5YF2 137655402 IC50 = 7700 nM T57392 CSRK73 137655508 IC50 > 100000 nM T57392 C17LIA 137655641 IC50 > 33000 nM T57392 CRY40J 137655938 IC50 = 330 nM T57392 C1OXG8 137655944 IC50 > 10000 nM T57392 C29UVL 137656780 IC50 = 197 nM T57392 C8DT1W 137657247 IC50 = 498 nM T57392 C2BGF3 137657547 IC50 = 120 nM T57392 CB61UY 137658460 IC50 = 18000 nM T57392 CG96FH 137658637 IC50 > 10000 nM T57392 C1R7UP 137658901 IC50 = 538 nM T57392 CKVH89 137658916 IC50 = 1900 nM T57392 CJ8L1W 137659170 IC50 = 17200 nM T57392 CA4MT5 137661210 IC50 = 33490 nM T57392 C96QPV 137662004 IC50 > 5000 nM T57392 CSEZ59 137662026 IC50 = 524 nM T57392 C6KYD7 137700754 IC50 > 10000 nM T57392 CJC95O 138319684 IC50 > 50000 nM T57392 CMP8U3 138376515 IC50 > 10000 nM T57392 CE79SV 138377584 IC50 > 50000 nM T57392 CKDZ26 138504497 IC50 > 30000 nM T57392 C1XSH7 138594194 IC50 > 10000 nM T57392 CG4RO6 138632227 IC50 > 18000 nM T57392 CHT39X 138632268 IC50 > 18000 nM T57392 CVB6L2 138632650 IC50 > 18000 nM T57392 CN9R4A 138691364 IC50 = 7470 nM T57392 CI9YB7 138753112 IC50 > 50000 nM T57392 CJA5H2 138756812 IC50 >= 20000 nM T57392 CD29IP 139507088 IC50 > 10000 nM T57392 CF8LN1 139582020 IC50 > 30000 nM T57392 CI1D9F 139600335 IC50 > 100000 nM T57392 CG2NH6 139600336 IC50 > 20000 nM T57392 C0HN5J 139600337 IC50 > 20000 nM T57392 CGA12N 141473855 IC50 = 38120 nM T57392 C2YC6F 141473885 IC50 = 24070 nM T57392 C9JSZ2 141529337 IC50 > 10000 nM T57392 CSE1D2 141529338 IC50 > 10000 nM T57392 C43LDR 141730928 IC50 > 50000 nM T57392 C06ZBJ 142416740 IC50 > 20000 nM T57392 C9J1ZO 142416754 IC50 = 540 nM T57392 C58KQF 142416884 IC50 = 81 nM T57392 C68OXK 142416914 IC50 = 110 nM T57392 C7C3MK 142416935 IC50 > 20000 nM T57392 CO7DK2 142416967 IC50 = 760 nM T57392 C1UCX0 144953608 IC50 > 10000 nM T57392 C9GRB2 144953612 IC50 > 10000 nM T57392 CV4X5P 144953614 IC50 > 10000 nM T57392 C1W8QR 145865307 IC50 > 50000 nM T57392 C9ISH6 145925685 IC50 > 20000 nM T57392 CVND41 145949156 IC50 = 1400 nM T57392 CF1MH2 145949267 IC50 > 30000 nM T57392 CI14LP 145949343 IC50 = 110 nM T57392 CXJ07F 145949470 IC50 = 10000 nM T57392 C8KA6P 145949486 IC50 = 2960 nM T57392 CA0B3D 145949907 IC50 > 20000 nM T57392 C7W9ZT 145949949 IC50 > 20000 nM T57392 CI3V6Y 145950358 IC50 = 2400 nM T57392 COG04E 145950432 IC50 = 190 nM T57392 CAWU95 145950510 IC50 = 8130 nM T57392 CLZ54T 145950740 IC50 = 2800 nM T57392 CL2OR1 145950976 IC50 > 20000 nM T57392 C4FM3C 145951105 IC50 = 6600 nM T57392 CLV0G6 145951167 IC50 = 21000 nM T57392 C2M8PI 145951236 IC50 > 20000 nM T57392 CH0K8V 145951521 IC50 > 10000 nM T57392 C3OMF2 145951963 IC50 = 140 nM T57392 CG5OW3 145951998 IC50 = 14000 nM T57392 CEB71V 145952023 IC50 > 30000 nM T57392 C4LJV9 145952024 IC50 = 12000 nM T57392 C1QA6W 145952070 IC50 = 3000 nM T57392 CC7IP8 145952109 IC50 = 4600 nM T57392 C3E5BK 145952508 IC50 > 10000 nM T57392 CC4K9F 145952601 IC50 > 20000 nM T57392 C0RGQ7 145952699 IC50 > 10000 nM T57392 CGW92C 145952721 IC50 = 2140 nM T57392 C2FXL5 145952723 IC50 = 508 nM T57392 C9D5MZ 145952745 IC50 > 50000 nM T57392 CRN85T 145952991 IC50 > 25000 nM T57392 CER83S 145953040 IC50 > 20000 nM T57392 CA7W2O 145953059 IC50 = 1700 nM T57392 C1A4CH 145953177 IC50 = 6090 nM T57392 COZ1F4 145953325 IC50 > 20000 nM T57392 C09WNF 145953342 IC50 = 4210 nM T57392 CEJ26X 145953403 IC50 = 6040 nM T57392 CS21ZB 145953739 IC50 = 5140 nM T57392 C5LB7M 145953999 IC50 = 12000 nM T57392 CW9I0R 145954143 IC50 > 10000 nM T57392 CPW52X 145954567 IC50 = 180 nM T57392 CN5L4K 145954640 IC50 = 3600 nM T57392 C59AVT 145954818 IC50 > 20000 nM T57392 C4P6MT 145954878 IC50 = 2520 nM T57392 CWA8H2 145955288 IC50 > 30000 nM T57392 CQ5SN1 145955289 IC50 > 50000 nM T57392 CK0S1G 145955694 IC50 > 20000 nM T57392 CE03RK 145955745 IC50 = 8450 nM T57392 CF6T7G 145955884 IC50 = 8570 nM T57392 C0HN4S 145955917 IC50 = 12000 nM T57392 C8Y4VT 145956312 IC50 > 20000 nM T57392 C4G6XJ 145956824 IC50 = 270 nM T57392 C7N6CA 145956935 IC50 > 50000 nM T57392 CBFU43 145957229 IC50 = 4500 nM T57392 CQ0JP4 145957239 IC50 > 20000 nM T57392 CK94HO 145957365 IC50 = 1870 nM T57392 C70LMY 145957553 IC50 > 20000 nM T57392 C20EDK 145957568 IC50 = 16000 nM T57392 CFZJ34 145957574 IC50 > 19952.62 nM T57392 CB2K0W 145957599 IC50 = 11000 nM T57392 C3B0YE 145957778 IC50 = 3900 nM T57392 CID3G5 145958087 IC50 > 50000 nM T57392 C8WZY3 145958093 IC50 = 1430 nM T57392 CXHM49 145958111 IC50 < 27 nM T57392 CBC1T9 145958296 IC50 = 88 nM T57392 C3TX8O 145958528 IC50 = 30 nM T57392 CM8U9A 145958674 IC50 = 3000 nM T57392 CT3U1A 145958698 IC50 = 6480 nM T57392 CBF54O 145958967 IC50 = 12000 nM T57392 CB5XW7 145959080 IC50 = 850 nM T57392 CH47WN 145959135 IC50 = 470 nM T57392 CW8M0I 145959142 IC50 > 20000 nM T57392 CLS3W5 145959177 IC50 > 25000 nM T57392 C8DH5F 145959814 IC50 = 1040 nM T57392 C5Z9US 145959844 IC50 = 5600 nM T57392 CLJE41 145959897 IC50 = 12000 nM T57392 CW1GO5 145960043 IC50 = 5000 nM T57392 CUD9E6 145960079 IC50 > 20000 nM T57392 CI8Q2V 145960175 IC50 = 59 nM T57392 C3F8XM 145960247 IC50 > 20000 nM T57392 CDKY72 145960338 IC50 = 8200 nM T57392 CT6OH1 145960389 IC50 > 50000 nM T57392 CZ83QK 145960490 IC50 > 50000 nM T57392 C0WB6J 145960881 IC50 > 20000 nM T57392 C5ZD1H 145961500 IC50 > 30000 nM T57392 CD01PX 145961863 IC50 = 4140 nM T57392 C42PLT 145962320 IC50 = 27200 nM T57392 CDY47R 145962388 IC50 > 50000 nM T57392 CQ2TN4 145962919 IC50 > 30000 nM T57392 CKLA91 145962920 IC50 = 2700 nM T57392 C64OLM 145963140 IC50 > 20000 nM T57392 CU8Y2C 145963537 IC50 = 6650 nM T57392 C62MVS 145964029 IC50 = 42600 nM T57392 CFAK41 145964101 IC50 = 7700 nM T57392 C2IM3V 145964416 IC50 = 4400 nM T57392 CRZ5T1 145964880 IC50 = 6600 nM T57392 C7SK5V 145965195 IC50 = 5700 nM T57392 CSK8Y1 145965486 IC50 = 3000 nM T57392 C4P7UD 145965756 IC50 = 14100 nM T57392 C42FZC 145966011 IC50 > 20000 nM T57392 C2MS3R 145966170 IC50 >= 30000 nM T57392 CRS65V 145966585 IC50 > 10000 nM T57392 CPH9E3 145967023 IC50 = 24000 nM T57392 CW02FZ 145967133 IC50 > 10000 nM T57392 CC0QA2 145967606 IC50 > 20000 nM T57392 C19IVD 145967885 IC50 > 20000 nM T57392 CX42BV 145968371 IC50 > 50000 nM T57392 CU6RH3 145968879 IC50 > 50000 nM T57392 CJUK65 145968931 IC50 > 10000 nM T57392 CCB21N 145969176 IC50 = 5600 nM T57392 C4HF5M 145969366 IC50 = 18000 nM T57392 C94URS 145969597 IC50 = 18000 nM T57392 C2S8DE 145969909 IC50 > 20000 nM T57392 CI3O2K 145970611 IC50 > 20000 nM T57392 C6CD4Z 145970793 IC50 > 20000 nM T57392 CS5U3M 145970807 IC50 > 20000 nM T57392 CND2K7 145971189 IC50 > 20000 nM T57392 CMI45E 145971507 IC50 = 12000 nM T57392 CXF9E7 145972420 IC50 = 760 nM T57392 CU13IP 145972573 IC50 > 10000 nM T57392 CP7LW2 145973146 IC50 = 5720 nM T57392 CV9OM2 145973260 IC50 > 10000 nM T57392 C8RFM3 145973261 IC50 > 20000 nM T57392 C8OSM0 145973345 IC50 > 20000 nM T57392 C6OI3K 145973962 IC50 > 10000 nM T57392 C4XZ1W 145973987 IC50 = 4500 nM T57392 C56HYE 145974067 IC50 = 20000 nM T57392 C54QHK 145974080 IC50 = 14200 nM T57392 CJN96Q 145974556 IC50 = 6500 nM T57392 CGWM29 145974840 IC50 = 21100 nM T57392 CAU82Y 145975252 IC50 > 10000 nM T57392 CSBQ67 145975261 IC50 > 10000 nM T57392 CUZ47S 145975654 IC50 > 10000 nM T57392 CQ2H6F 145976125 IC50 > 10000 nM T57392 CUV49K 145977796 IC50 = 22000 nM T57392 C4XV7J 145978553 IC50 > 10000 nM T57392 C3S0UI 145978581 IC50 = 10800 nM T57392 CWA6L3 145981037 IC50 = 1600 nM T57392 CGA83C 145981271 IC50 > 10000 nM T57392 CJ35DM 145984299 IC50 > 100000 nM T57392 C4HAP0 145984727 IC50 = 15100 nM T57392 C5R6BS 145987142 IC50 > 10000 nM T57392 C7O1PF 145987480 IC50 > 20000 nM T57392 C81LEH 145987485 IC50 > 20000 nM T57392 CMRQ02 145987862 IC50 = 1400 nM T57392 C7GK3H 145990715 IC50 > 100000 nM T57392 CE1L5T 145992719 IC50 > 20000 nM T57392 CMIH10 145993513 IC50 = 200 nM T57392 C8X2IT 145996536 IC50 > 50000 nM T57392 CHJ79V 145997874 IC50 > 10000 nM T57392 CAU3Z1 146020618 IC50 > 40000 nM T57392 CZE16B 146026197 IC50 > 50000 nM T57392 C7F6SU 146047134 IC50 > 200000 nM T57392 CBRE71 146047136 IC50 > 20000 nM T57392 C2RJ1U 146176418 IC50 > 50000 nM T57392 CS54CM 146433251 IC50 > 40000 nM T57392 CGO5C4 146433253 IC50 > 40000 nM T57392 C61LGO 146433463 IC50 > 40000 nM T57392 C4OSN5 146433538 IC50 > 40000 nM T57392 CN2MA4 146433574 IC50 > 40000 nM T57392 C5ZOJ3 146680920 IC50 > 100000 nM T57392 C9YJZ5 147180858 IC50 = 23800 nM T57392 CUAY08 148018738 IC50 > 10000 nM T57392 CQK39B 149491764 IC50 > 10000 nM T57392 C1ZX5D 149494192 IC50 > 10000 nM T57392 CL6T4P 149986651 IC50 > 20000 nM T57392 CTI5R1 151961601 IC50 > 20000 nM T57392 CC3ME1 152131905 IC50 > 20000 nM T57392 C36ISR 153434865 IC50 > 10000 nM T57392 CG5IF7 154701259 IC50 > 1000 nM T57392 C2J9YV 154727580 IC50 = 299000 nM T57392 CZE1S5 155126870 IC50 > 50000 nM T57392 CI6EB5 155126882 IC50 > 50000 nM T57392 CF2CU8 155510758 IC50 > 30000 nM T57392 C7ZE5Q 155511547 IC50 = 80 nM T57392 CXW4J6 155512369 IC50 = 5400 nM T57392 CQ83KZ 155512662 IC50 > 10000 nM T57392 C5M6NS 155513226 IC50 > 27000 nM T57392 C8SW9I 155513332 IC50 = 6000 nM T57392 CG73TZ 155513551 IC50 > 20000 nM T57392 C17RIB 155513592 IC50 > 20000 nM T57392 CPE58H 155514125 IC50 > 20000 nM T57392 CZUP45 155514353 IC50 > 30000 nM T57392 CD53LC 155514863 IC50 = 10000 nM T57392 C9HG0U 155515457 IC50 > 20000 nM T57392 CMZ4Q7 155515478 IC50 > 25000 nM T57392 CDV4Z6 155515709 IC50 = 1710000 nM T57392 C7OF4C 155516118 IC50 = 8400 nM T57392 CCJ14L 155516448 IC50 = 4510 nM T57392 C49INQ 155516757 IC50 > 50000 nM T57392 CA3K9P 155517032 IC50 < 10000 nM T57392 CQ52LM 155518361 IC50 > 20000 nM T57392 CRD79Z 155518589 IC50 < 10000 nM T57392 C30SPO 155518654 IC50 > 50000 nM T57392 C28HEF 155519544 IC50 > 100000 nM T57392 C0KLD8 155519559 IC50 > 100000 nM T57392 C1U3CL 155520250 IC50 > 20000 nM T57392 CF19DM 155521087 IC50 > 30000 nM T57392 CI9U3X 155521508 IC50 > 20000 nM T57392 CK7RM1 155521671 IC50 >= 20000 nM T57392 C0ZXV4 155522886 IC50 < 10000 nM T57392 CC5GO1 155523088 IC50 > 50000 nM T57392 C2LO4Y 155523731 IC50 < 10000 nM T57392 C3LC2H 155523754 IC50 > 20000 nM T57392 C12KNB 155523817 IC50 = 240 nM T57392 CYI71L 155523951 IC50 > 40000 nM T57392 CTU67Z 155524559 IC50 > 100000 nM T57392 CFM45O 155524794 IC50 = 12700 nM T57392 CG71WI 155525128 IC50 < 10000 nM T57392 CI31SP 155527821 IC50 = 11600 nM T57392 C05QTC 155528035 IC50 = 10000 nM T57392 C0B2NV 155528644 IC50 > 27000 nM T57392 C5QA2B 155529241 IC50 < 10000 nM T57392 C9U8FN 155529326 IC50 > 50000 nM T57392 C7SEX2 155529894 IC50 = 43200 nM T57392 C4F7WU 155530183 IC50 = 32580 nM T57392 CK5X2E 155530190 IC50 > 20000 nM T57392 CQ6F7O 155530369 IC50 < 10000 nM T57392 CQD26H 155530468 IC50 > 20000 nM T57392 CFL61W 155532250 IC50 = 16000 nM T57392 CH62TN 155532900 IC50 = 4000 nM T57392 C63HSA 155534748 IC50 > 50000 nM T57392 CTH8B9 155535743 IC50 > 20000 nM T57392 CY97DN 155535886 IC50 > 20000 nM T57392 C7FVE8 155537034 IC50 = 27600 nM T57392 CM1BX0 155537411 IC50 > 20000 nM T57392 C8K3XJ 155537606 IC50 = 17800 nM T57392 CM3PB2 155537682 IC50 < 10000 nM T57392 CCO96S 155538113 IC50 > 100000 nM T57392 C6KX1G 155538348 IC50 > 20000 nM T57392 CDU52V 155538567 IC50 = 90 nM T57392 CUS3I9 155538644 IC50 < 10000 nM T57392 C1FZY9 155539610 IC50 = 19100 nM T57392 CGH8T5 155540333 IC50 > 10000 nM T57392 CB43YR 155540395 IC50 > 40000 nM T57392 C5T9KE 155542416 IC50 > 50000 nM T57392 C1SY0G 155543154 IC50 > 27000 nM T57392 CNH46F 155543687 IC50 > 40000 nM T57392 CQ6D2C 155547369 IC50 > 25000 nM T57392 CRY3A2 155548898 IC50 > 30000 nM T57392 CH25ZD 155549064 IC50 > 50000 nM T57392 CJD38X 155549583 IC50 > 25000 nM T57392 C08YOZ 155549638 IC50 > 20000 nM T57392 CD4PW8 155550069 IC50 > 20000 nM T57392 CHDG36 155550819 IC50 > 25000 nM T57392 CGDS14 155551776 IC50 > 20000 nM T57392 C7JH8N 155552861 IC50 > 20000 nM T57392 CUH7R2 155553391 IC50 > 10000 nM T57392 C7JCS2 155553955 IC50 > 25000 nM T57392 C7N5HA 155554052 IC50 > 50000 nM T57392 C3J2YD 155554863 IC50 = 2000 nM T57392 C3Z4QS 155554969 IC50 > 20000 nM T57392 C8Q2FG 155555556 IC50 > 20000 nM T57392 C09FGY 155555863 IC50 < 10000 nM T57392 CIK75H 155556042 IC50 > 25000 nM T57392 C3WT2Q 155556441 IC50 > 50000 nM T57392 C9H1VK 155556442 IC50 > 50000 nM T57392 CQB48L 155556931 IC50 > 50000 nM T57392 CFS63H 155557182 IC50 > 27000 nM T57392 CNH27R 155557555 IC50 > 20000 nM T57392 C4HPK2 155558743 IC50 > 25000 nM T57392 CKZT21 155559364 IC50 > 20000 nM T57392 CEF9N6 155560028 IC50 < 10000 nM T57392 CW2N7D 155560551 IC50 = 3000 nM T57392 C1NVA6 155560651 IC50 > 30000 nM T57392 CF4LM6 155560880 IC50 > 25000 nM T57392 CM7ZG9 155561160 IC50 < 10000 nM T57392 C9HIU5 155561551 IC50 < 10000 nM T57392 C1MW3L 155561646 IC50 > 40000 nM T57392 CALB48 155561861 IC50 > 10000 nM T57392 CL3A2S 155562076 IC50 = 700 nM T57392 CKX10W 155562129 IC50 = 49600 nM T57392 C6T2RV 155562253 IC50 < 10000 nM T57392 CCOD50 155562467 IC50 > 30000 nM T57392 CFVB79 155562854 IC50 = 50000 nM T57392 CG95WV 155563831 IC50 > 20000 nM T57392 CWOE21 155564042 IC50 > 30000 nM T57392 CMK03D 155564568 IC50 < 10000 nM T57392 CC5FE7 155564581 IC50 > 50000 nM T57392 CIBA72 155564665 IC50 > 50000 nM T57392 C37BGO 155567311 IC50 > 30000 nM T57392 C16AQH 155567592 IC50 = 4800 nM T57392 CK9N0Z 155567885 IC50 > 10000 nM T57392 CMC2A9 155568311 IC50 > 50000 nM T57392 CYIU14 16750228 IC50 > 10000 nM T57392 CI67WG 16750292 IC50 > 10000 nM T57392 C9JX2G 53363150 IC50 > 10000 nM T57392 CU76JB 53363338 IC50 > 10000 nM T57392 CKYJ21 76283430 IC50 > 20000 nM T57392 CIJ3N0 76283682 IC50 > 30000 nM T57392 D00AEX 44341439 IC50 = 1000 nM T57392 D00AWM 9826520 IC50 > 10000000 nM T57392 D00EMF 3644637 IC50 > 100000 nM T57392 D00GEE 92766 Ki = 80 nM T57392 D00GOQ 44575384 IC50 > 100000 nM T57392 D00PYW 44341256 IC50 = 399 nM T57392 D00TOF 193042 IC50 = 17500 nM T57392 D00XDG 11708263 IC50 > 30000 nM T57392 D00YNA 25093374 IC50 > 4000 nM T57392 D01ARE 44388719 IC50 = 14400 nM T57392 D01DAU 24825518 IC50 = 644 nM T57392 D01FBL 442835 IC50 = 95700 nM T57392 D01JFF 44191096 IC50 > 30000 nM T57392 D01JPJ 66731056 IC50 > 10000 nM T57392 D01JXM 46222048 IC50 = 680 nM T57392 D01RZP 25192621 IC50 = 1500 nM T57392 D01SHR 44593693 IC50 = 1600 nM T57392 D01UYI 5281607 IC50 > 50000 nM T57392 D01YWE 25207521 IC50 > 10000 nM T57392 D02BGR 9949648 IC50 > 100000 nM T57392 D02DCM 44230874 IC50 = 100 nM T57392 D02DEF 49765871 IC50 > 30000 nM T57392 D02DTR 44341278 IC50 = 1300 nM T57392 D02EAP 11993867 Ki = 38400 nM T57392 D02GFK 25034431 IC50 = 11100 nM T57392 D02HSP 44575401 IC50 > 100000 nM T57392 D02KZD 71598521 IC50 = 26000 nM T57392 D02TSN 46244454 IC50 > 10000 nM T57392 D03KXT 44341260 IC50 = 1040 nM T57392 D03NMM 46843035 IC50 > 30000 nM T57392 D03SAV 3082718 IC50 = 26 nM T57392 D03YHZ 25147692 IC50 = 50000 nM T57392 D05FNN 100606 IC50 = 699000 nM T57392 D05KIF 13916150 IC50 > 100000 nM T57392 D05LKO 44414722 IC50 = 20000 nM T57392 D05MSG 44593666 IC50 = 1600 nM T57392 D05NWH 443390 IC50 = 21000 nM T57392 D05VQJ 25147749 IC50 = 400 nM T57392 D05XGR 6918647 IC50 = 11000 nM T57392 D06CWR 24754344 IC50 = 33110 nM T57392 D06EMC 11392888 IC50 > 30000 nM T57392 D06HOI 44249821 IC50 > 200000 nM T57392 D06MBD 11176403 IC50 = 6780 nM T57392 D06MLU 332806 IC50 > 100000 nM T57392 D06QFO 11332763 Ki = 5700 nM T57392 D06TRS 23646069 Ki = 48000 nM T57392 D06UEP 17027464 IC50 > 25000 nM T57392 D06VDN 443391 IC50 > 100000 nM T57392 D07ADX 54764565 IC50 > 30000 nM T57392 D07ANY 1367 IC50 = 10500 nM T57392 D07GCA 11514705 IC50 > 10000 nM T57392 D07VHB 11321889 IC50 = 460 nM T57392 D07WLT 25180108 IC50 = 171000 nM T57392 D08BOH 192827 IC50 > 100000 nM T57392 D08EKQ 46890532 IC50 = 1400 nM T57392 D08IDC 24827305 IC50 > 25000 nM T57392 D08QPU 72737723 IC50 = 12000 nM T57392 D08UWZ 16725047 IC50 > 40000 nM T57392 D08ZYC 11595431 IC50 > 33000 nM T57392 D09CPC 13728862 IC50 = 171000 nM T57392 D09FIC 46890395 IC50 = 3000 nM T57392 D09PTP 57325421 IC50 > 10000 nM T57392 D09VMS 44575398 IC50 > 100000 nM T57392 D09ZPN 135416394 IC50 > 100000 nM T57392 D0A0GU 44247568 IC50 > 10000 nM T57392 D0A1SJ 44575400 IC50 = 87900 nM T57392 D0AS0V 10141 IC50 > 10000 nM T57392 D0B0LC 44341428 IC50 = 1040 nM T57392 D0B2ZB 3013841 IC50 > 100000 nM T57392 D0BD6A 10278617 IC50 > 10000 nM T57392 D0BU8W 44219611 IC50 > 100000 nM T57392 D0BV3B 16214871 IC50 > 30000 nM T57392 D0BW0V 44589528 IC50 = 3100 nM T57392 D0C4XQ 44316307 IC50 = 1210 nM T57392 D0C7PK 3123920 IC50 = 18000 nM T57392 D0DA1E 23642319 IC50 = 2000 nM T57392 D0DY5G 443389 IC50 = 110 nM T57392 D0F5AQ 49798218 IC50 = 60 nM T57392 D0F5EI 10017019 IC50 > 10000 nM T57392 D0FF0Z 24825516 IC50 = 488 nM T57392 D0FQ1Z 101711 Ki = 1600 nM T57392 D0G6BJ 24802842 IC50 = 3000 nM T57392 D0G8KT 44409490 IC50 = 15000 nM T57392 D0G8UA 46890321 IC50 > 30000 nM T57392 D0G9WP 18407230 IC50 < 200000 nM T57392 D0GG2J 46890492 IC50 = 3100 nM T57392 D0H1OK 11562302 IC50 = 33000 nM T57392 D0H8XV 12963076 IC50 = 32500 nM T57392 D0I2UC 44230733 IC50 = 100 nM T57392 D0I7GE 11790 IC50 > 10000 nM T57392 D0IM5E 11450263 IC50 = 3400 nM T57392 D0IO0I 6474893 IC50 = 600 nM T57392 D0IO8J 3025961 IC50 > 100000 nM T57392 D0J0TP 9917862 IC50 > 30000 nM T57392 D0J1IE 11993873 Ki = 64500 nM T57392 D0J1QT 44473100 IC50 > 40000 nM T57392 D0J2YB 23631116 IC50 = 13000 nM T57392 D0J4CB 24803184 IC50 = 8000 nM T57392 D0J6RQ 6437306 IC50 = 2000 nM T57392 D0J9SO 11964445 IC50 = 60 nM T57392 D0K3EW 49799108 IC50 = 3000 nM T57392 D0K4LS 10691533 IC50 = 82700 nM T57392 D0L2WP 46225540 IC50 = 5000 nM T57392 D0L9YP 44254503 IC50 = 440 nM T57392 D0M0IQ 11210706 IC50 = 12900 nM T57392 D0M0KX 25192477 IC50 = 1500 nM T57392 D0M4SY 135440466 IC50 > 40000 nM T57392 D0M7SY 9910352 IC50 = 800 nM T57392 D0N2KU 44517677 IC50 = 15100 nM T57392 D0N4LR 53469448 IC50 = 23000 nM T57392 D0NC3P 117443 IC50 = 35500 nM T57392 D0NM0P 25093389 IC50 > 4000 nM T57392 D0O1HH 11263510 Ki = 60500 nM T57392 D0O8WT 10338547 IC50 > 30000 nM T57392 D0P0IE 10205 IC50 > 10000 nM T57392 D0P2DU 65775 Ki = 4.8 nM T57392 D0P8PK 10192730 IC50 = 32560 nM T57392 D0PC5A 44243144 IC50 > 10000 nM T57392 D0QH6F 8931837 IC50 = 10000 nM T57392 D0R0IB 56587994 IC50 > 30000 nM T57392 D0R0TW 11964036 IC50 > 10000 nM T57392 D0R2TW 10238338 IC50 > 100000 nM T57392 D0S1XC 25224941 IC50 = 3400 nM T57392 D0S6GE 5327067 IC50 = 25000 nM T57392 D0S6NP 5280862 IC50 = 4630 nM T57392 D0S9CI 11989776 IC50 > 30000 nM T57392 D0SE3C 56661208 IC50 = 150 nM T57392 D0T4AC 11259008 IC50 > 100000 nM T57392 D0U7BJ 44341234 IC50 = 620 nM T57392 D0U7OD 16043230 IC50 = 30000 nM T57392 D0V0YM 24871527 IC50 = 6000 nM T57392 D0V2QH 24894072 IC50 = 15490 nM T57392 D0V3ZG 25192022 IC50 > 7500 nM T57392 D0V4EX 54760053 IC50 > 40000 nM T57392 D0VD5O 11148236 Ki > 400000 nM T57392 D0W3XD 16049828 IC50 > 30000 nM T57392 D0W8CA 46846313 IC50 = 100 nM T57392 D0X3CF 442879 IC50 = 26500 nM T57392 D0X4DE 44409554 IC50 = 210 nM T57392 D0Y2RL 25192475 IC50 = 1500 nM T57392 D0YM4A 22319604 IC50 > 10000 nM T57392 D0YP4A 11993866 Ki = 700 nM T57392 D0YQ8U 11993871 Ki = 14800 nM T57392 D0YQ8V 46236221 IC50 > 30000 nM T57392 D0ZC3Q 44230732 IC50 = 500 nM T57392 D0ZY7X 697226 IC50 = 4200 nM T57392 D0ZZ2L 56678302 IC50 = 260 nM T17048 D07VLY 31703 IC50 = 1000 nM T17048 D0B7EB 36462 IC50 = 28200 nM T17048 D0G9YH 2179 IC50 = 9940 nM T17048 D0K8KX 5280343 IC50 = 6.9 ug.mL-1 T17048 D0O1WX 2764 IC50 = 153600 nM T17048 D0Q0PR 54675769 IC50 > 256000 nM T17048 D0R3JB 4212 IC50 = 5300 nM T17048 D08BXT 1102 IC50 > 1000000 nM T17048 D09YDM 24360 IC50 > 300000 nM T17048 D0L4FS 5280961 IC50 = 30 ug.mL-1 T17048 D00VZF 4990817 IC50 = 26000 nM T17048 D04ZLJ 72116 IC50 = 7300 nM T17048 D0LD9S 1103 IC50 > 1000000 nM T17048 D0OH5V 59916 IC50 = 4600 nM T17048 CU6P5W 35296 IC50 > 1000000 nM T17048 CEC4M7 73104 IC50 = 25 ug.mL-1 T17048 CKH0W1 73170 IC50 > 250000 nM T17048 C80OQM 94303 IC50 = 18600 nM T17048 CA4IO8 115150 IC50 = 13900 nM T17048 CVB5T2 127748 IC50 = 32000 nM T17048 CQ9BN3 189219 IC50 = 1376 nM T17048 C5U4SA 372621 IC50 > 500000 nM T17048 CF7AE4 400717 IC50 = 700 nM T17048 CNJ0Q6 400718 IC50 = 60 nM T17048 CCK68G 441921 IC50 > 250000 nM T17048 CYMH94 471008 IC50 = 17000 nM T17048 C6N9OU 617467 IC50 > 1000000 nM T17048 CH76XU 637031 IC50 = 75700 nM T17048 CK9ES8 943044 IC50 = 85000 nM T17048 C20VLU 1319814 IC50 > 1000000 nM T17048 CB7JW9 1332897 IC50 > 1000000 nM T17048 C5XL1M 1385849 IC50 = 139000 nM T17048 CAF2O7 1554842 IC50 = 229000 nM T17048 C8V1TW 2723942 IC50 = 26950 nM T17048 CKS4I5 2818525 IC50 > 1000000 nM T17048 CAP70Y 2826719 IC50 > 1000000 nM T17048 CKD72T 3083848 IC50 = 404000 nM T17048 CJG60Z 3332833 IC50 > 1000000 nM T17048 COY89G 3738100 IC50 = 25800 nM T17048 CRU5O7 3758536 IC50 > 1000000 nM T17048 C5JRO9 4159286 IC50 > 1000000 nM T17048 CCZ53E 4245203 IC50 > 1000000 nM T17048 CF0GI2 4289636 IC50 > 1000000 nM T17048 C4E0LT 4294777 IC50 = 44000 nM T17048 CI1H5A 5098538 IC50 > 1000000 nM T17048 C0WXP5 5284649 IC50 = 43.7 ug.mL-1 T17048 CI9TO8 5307536 IC50 = 680 nM T17048 C13OPQ 5352088 IC50 = 101200 nM T17048 C7AV1K 5371064 IC50 > 100000 nM T17048 C02JQT 5375900 IC50 > 100000 nM T17048 CX3EZ6 5382559 IC50 > 100000 nM T17048 C8HSR7 5488193 IC50 >= 100000 nM T17048 C2KO9P 5711011 IC50 = 76000 nM T17048 C8DB1Y 5920829 IC50 = 79000 nM T17048 CK4R6S 5996579 IC50 = 92000 nM T17048 C4LY8R 6892730 IC50 > 100000 nM T17048 CVY36D 7694997 IC50 > 100000 nM T17048 C2TA8R 7728685 IC50 = 94000 nM T17048 CJ3Z6F 9208033 IC50 > 1000000 nM T17048 C4UHE7 9577310 IC50 > 100000 nM T17048 C9P5KJ 9602564 IC50 > 100000 nM T17048 CH39YU 9637541 IC50 = 1910 nM T17048 CX5CR4 9831582 IC50 = 24100 nM T17048 CQX6Y4 9837937 IC50 > 400000 nM T17048 CLI8Z3 9898279 IC50 > 250000 nM T17048 CF0O4M 9918692 IC50 > 250000 nM T17048 CQRD02 9927270 IC50 = 1 ug.mL-1 T17048 C8ME5O 10260430 IC50 = 2 ug.mL-1 T17048 CH6L2I 10318315 IC50 = 168900 nM T17048 C9UF8K 10676329 IC50 > 200000 nM T17048 CI4AB2 10741986 IC50 > 100000 nM T17048 C0B1OM 10747298 IC50 > 200000 nM T17048 CA2S8I 10933039 IC50 > 400000 nM T17048 CE38LT 10961552 IC50 = 50400 nM T17048 CS12LC 11049543 IC50 = 67300 nM T17048 COQ35J 11188178 IC50 = 29560 nM T17048 C8OH4C 11300612 IC50 > 1000000 nM T17048 CCJM42 11313757 IC50 = 16740 nM T17048 CO9K4F 11406001 IC50 = 18040 nM T17048 CM6SF2 11414937 IC50 = 120000 nM T17048 CE74PN 11425952 IC50 = 67860 nM T17048 CB5D6Y 11474949 IC50 = 7500 nM T17048 CQR90J 11623140 IC50 > 400000 nM T17048 CO0SR8 11629881 IC50 = 55600 nM T17048 CS80WY 11679800 IC50 > 250000 nM T17048 C9HQ4Z 11776102 IC50 > 100000 nM T17048 CK1J8Q 11779019 IC50 = 12.5 ug.mL-1 T17048 CER3U0 11788101 IC50 > 250000 nM T17048 C14PRE 11799152 IC50 = 8900 nM T17048 CARZ73 11975877 IC50 = 240000 nM T17048 C7JYP0 12133302 IC50 = 4600 nM T17048 CN8RP5 12306720 IC50 = 35000 nM T17048 CEC68V 12912322 IC50 > 250000 nM T17048 CK3MX1 12912363 IC50 > 250000 nM T17048 CVN35P 13385680 IC50 = 2090 nM T17048 C2Y0IW 13495619 IC50 = 1060 nM T17048 C21WBU 14037821 IC50 = 125 nM T17048 C5J0PE 14167253 IC50 > 200000 nM T17048 C7CLT5 14167260 IC50 = 38700 nM T17048 CRHQ70 14194006 IC50 > 250000 nM T17048 C5P7AC 14194010 IC50 > 250000 nM T17048 CHD3G6 14203214 IC50 > 400000 nM T17048 CM0CG1 14316872 IC50 = 250000 nM T17048 CRST54 14316873 IC50 = 3900 nM T17048 C3TGM9 14380944 IC50 = 76 nM T17048 C23ANM 14804068 IC50 > 400000 nM T17048 CQR46S 15068049 IC50 = 1950 nM T17048 CJ8NX1 16048967 IC50 = 32000 nM T17048 CAEZ10 17478154 IC50 > 1000000 nM T17048 C5AUX1 17506081 IC50 > 1000000 nM T17048 COB0W1 17562978 IC50 > 1000000 nM T17048 C7F6HP 19420351 IC50 > 1000000 nM T17048 CTA53Z 21072872 IC50 = 28600 nM T17048 CP6D9H 21072873 IC50 = 55600 nM T17048 CA6P8H 21072874 IC50 = 52800 nM T17048 CN09HI 21072875 IC50 = 39000 nM T17048 CJY93K 21072876 IC50 = 43200 nM T17048 C03FLI 21072877 IC50 = 49000 nM T17048 CRI2B4 21072878 IC50 = 61500 nM T17048 CW3U7E 21072879 IC50 = 64800 nM T17048 C4FK9B 21072880 IC50 = 44400 nM T17048 CDG36B 21350957 IC50 > 400000 nM T17048 CGW4Q6 21580556 IC50 > 250000 nM T17048 CER14Y 21602071 IC50 = 42600 nM T17048 C74HBW 21606527 IC50 = 600000 nM T17048 C69EDW 21636448 IC50 > 250000 nM T17048 CAK48U 24939294 IC50 = 19400 nM T17048 CK5V4T 24970451 IC50 > 250000 nM T17048 CQ5V6L 25067849 IC50 = 550000 nM T17048 CQ7W8A 25067894 IC50 = 240000 nM T17048 C69QVI 25164720 IC50 = 25000 nM T17048 CPE1K9 25164921 IC50 = 50000 nM T17048 C1YHA2 25164923 IC50 = 42000 nM T17048 C0G8JQ 25165123 IC50 = 7000 nM T17048 CFO68D 25165124 IC50 = 25000 nM T17048 C6TI4Y 25165125 IC50 = 48000 nM T17048 CX40MO 25165319 IC50 = 22000 nM T17048 CUG78D 27213568 IC50 > 1000000 nM T17048 CHAM95 33499296 IC50 > 1000000 nM T17048 CG04EZ 39378450 IC50 = 65000 nM T17048 CJSG05 39794153 IC50 > 1000000 nM T17048 CJ28KY 39794232 IC50 > 1000000 nM T17048 C25SXL 39818372 IC50 > 1000000 nM T17048 CU23LJ 39997960 IC50 > 1000000 nM T17048 C5O3VE 40789334 IC50 > 1000000 nM T17048 CBN95G 44249746 IC50 = 1700 nM T17048 CHQD42 44249747 IC50 = 8400 nM T17048 C6RK3T 44338931 IC50 > 100000 nM T17048 CJPQ89 44338938 IC50 = 38000 nM T17048 C17RAS 44401260 IC50 > 400000 nM T17048 CWJL24 44401288 IC50 > 400000 nM T17048 CR3JN2 44401681 IC50 = 327000 nM T17048 CXCM26 44401682 IC50 = 272000 nM T17048 CT4K5F 44401784 IC50 > 400000 nM T17048 CUB96N 44401847 IC50 > 400000 nM T17048 C90WTK 44401922 IC50 = 63000 nM T17048 CAC38H 44401925 IC50 = 351000 nM T17048 CR7ZO4 44424826 IC50 = 37500 nM T17048 CI6T3F 44451937 IC50 = 33300 nM T17048 CB9M1J 44452368 IC50 = 29800 nM T17048 CI3DP0 44452369 IC50 = 54500 nM T17048 CNT3L9 44454668 IC50 = 19000 nM T17048 CBC86V 44454669 IC50 = 13000 nM T17048 CB4HR6 44456311 IC50 = 20490 nM T17048 C63WQJ 44456314 IC50 = 12270 nM T17048 CE73KZ 44456349 IC50 = 64340 nM T17048 CC57TE 44456350 IC50 = 15420 nM T17048 CTLC12 44456381 IC50 = 21200 nM T17048 CIAB35 44479228 IC50 > 250000 nM T17048 C0NL5G 44567396 IC50 = 7200 nM T17048 CT9FE8 44574831 IC50 = 40950 nM T17048 C2L6MX 44584555 IC50 > 250000 nM T17048 C5ODW8 44598780 IC50 = 6000 nM T17048 COHJ10 45028269 IC50 = 8000 nM T17048 CHK2I6 45028271 IC50 = 3000 nM T17048 CR98IM 45028272 IC50 = 12000 nM T17048 C1JD5G 45028273 IC50 = 10000 nM T17048 C1G2PX 45028274 IC50 = 18000 nM T17048 C3B9WD 45029396 IC50 > 100000 nM T17048 CA17OX 45029397 IC50 > 100000 nM T17048 C8N9BW 45381704 IC50 = 50000 nM T17048 C78ZFO 45481988 IC50 = 25000 nM T17048 CH24ZT 45481989 IC50 = 18000 nM T17048 CQA04W 46179700 IC50 > 1000000 nM T17048 CB3RD9 46179703 IC50 > 1000000 nM T17048 CL4PO2 46179760 IC50 > 1000000 nM T17048 C0S8XN 46179761 IC50 > 1000000 nM T17048 C0B4CK 46179762 IC50 > 1000000 nM T17048 C85COV 46179765 IC50 > 1000000 nM T17048 C2UDV0 46179812 IC50 > 1000000 nM T17048 CLF1W9 46179814 IC50 > 1000000 nM T17048 CPT2V4 46179869 IC50 > 1000000 nM T17048 C82KYI 46179870 IC50 > 1000000 nM T17048 C1PN9C 46224647 IC50 > 250000 nM T17048 C81QNL 46229825 IC50 = 114000 nM T17048 CNC12E 46887586 IC50 > 250000 nM T17048 CN49UH 46887587 IC50 > 250000 nM T17048 CQI2S5 46887678 IC50 > 250000 nM T17048 CPV4N6 46887679 IC50 > 250000 nM T17048 CR1JF6 46887680 IC50 > 250000 nM T17048 C6NPL9 46887682 IC50 > 250000 nM T17048 CN3KO1 46888244 IC50 > 250000 nM T17048 C4FOQ9 46888245 IC50 > 250000 nM T17048 C23BUR 46888246 IC50 > 250000 nM T17048 C10DYA 46888247 IC50 > 250000 nM T17048 CNF63K 46888248 IC50 > 250000 nM T17048 CX16CG 46888249 IC50 > 250000 nM T17048 C7Z8AK 46888250 IC50 > 250000 nM T17048 C6Z0OV 46888251 IC50 > 250000 nM T17048 CJEQ63 46888252 IC50 > 250000 nM T17048 CB36TZ 46888253 IC50 > 250000 nM T17048 C58XEI 46888254 IC50 > 250000 nM T17048 C1OMX0 46888255 IC50 > 250000 nM T17048 CUL8I2 46888256 IC50 > 250000 nM T17048 C3I1NG 46888257 IC50 > 250000 nM T17048 C8GOY7 46888258 IC50 > 250000 nM T17048 C38NOI 46888259 IC50 > 250000 nM T17048 CQP4R3 46888260 IC50 > 250000 nM T17048 CY6W1R 46888296 IC50 > 250000 nM T17048 C8NPJ6 46888298 IC50 > 250000 nM T17048 CJM78A 46888299 IC50 > 250000 nM T17048 C9O3GR 46888300 IC50 > 250000 nM T17048 CLN81T 46888301 IC50 > 250000 nM T17048 CQD47J 46888307 IC50 > 250000 nM T17048 CQ43PL 46888308 IC50 > 250000 nM T17048 CQ7H3G 46888311 IC50 > 250000 nM T17048 CR6TY2 46888312 IC50 > 250000 nM T17048 CR5SB4 46888313 IC50 > 250000 nM T17048 CK6YH8 46888320 IC50 > 250000 nM T17048 C4LXR1 46888321 IC50 > 250000 nM T17048 CLM5U7 46888322 IC50 > 250000 nM T17048 CTF0E5 46888323 IC50 > 250000 nM T17048 C06WJX 46888324 IC50 > 250000 nM T17048 C4XW3T 50907898 IC50 = 17000 nM T17048 C84JFQ 53248766 IC50 = 10400 nM T17048 CY8ME0 53361576 IC50 = 1880 nM T17048 CELQ84 53376152 IC50 = 1540 nM T17048 CILW42 53376258 IC50 = 4880 nM T17048 CWB54K 53380489 IC50 = 52660 nM T17048 C6C1JP 54210863 IC50 > 1000000 nM T17048 CIMR05 54578483 IC50 = 94100 nM T17048 CX58ZH 54578708 IC50 = 54600 nM T17048 C84WMD 54578709 IC50 = 219300 nM T17048 CK74GM 54579405 IC50 > 1000000 nM T17048 CY0WE3 54768945 IC50 = 485300 nM T17048 C0RFL5 54768946 IC50 > 1000000 nM T17048 C82FCG 54768947 IC50 = 72500 nM T17048 CJ67EC 54768949 IC50 = 146600 nM T17048 CXA98K 54768950 IC50 = 376700 nM T17048 C7XZ9Y 54769181 IC50 = 488300 nM T17048 C3YVZ9 54769182 IC50 = 358900 nM T17048 C96HPC 54769183 IC50 = 522000 nM T17048 C75WBG 54769184 IC50 = 528000 nM T17048 C48EJD 54769407 IC50 = 153400 nM T17048 C3J1KQ 54769408 IC50 = 485800 nM T17048 CQ08JC 54769410 IC50 > 1000000 nM T17048 CDL43S 54769411 IC50 = 234700 nM T17048 C19TGW 54769414 IC50 = 481000 nM T17048 C2VT4I 54769628 IC50 > 1000000 nM T17048 C3UQ8I 56659987 IC50 > 1000000 nM T17048 CLQ5N8 56680462 IC50 > 1000000 nM T17048 C3O8LT 56680463 IC50 > 1000000 nM T17048 C0SB1D 56682538 IC50 > 1000000 nM T17048 CY3EJ8 56683793 IC50 > 1000000 nM T17048 CM7Q3S 57401109 IC50 = 330000 nM T17048 C1C0VM 58160590 IC50 = 51600 nM T17048 CJ2HT1 60168004 IC50 = 3000 nM T17048 C0MT7I 60168005 IC50 = 15000 nM T17048 C8PBX5 60168006 IC50 = 5000 nM T17048 CV2R5U 66575905 IC50 > 256000 nM T17048 C9MLV8 67449276 IC50 > 256000 nM T17048 CMJ60D 67450057 IC50 > 256000 nM T17048 CQGK50 71459520 IC50 = 25000 nM T17048 C4U3MS 72201605 IC50 = 14500 nM T17048 CO7XG1 72201606 IC50 = 2100 nM T17048 C5HXU0 72203803 IC50 = 3000 nM T17048 CG24ZN 72203805 IC50 = 2000 nM T17048 CV1OD5 72206053 IC50 > 100000 nM T17048 CJD6N7 72206054 IC50 > 100000 nM T17048 C8C1YG 72206407 IC50 > 100000 nM T17048 CYS68B 72206408 IC50 > 100000 nM T17048 C37PKB 72375544 IC50 > 200000 nM T17048 CT48HB 72375652 IC50 = 149000 nM T17048 C0OIS7 72375653 IC50 > 200000 nM T17048 C0GQR3 72375654 IC50 > 200000 nM T17048 C3MG7F 72375655 IC50 > 200000 nM T17048 CU96NC 72375750 IC50 = 78900 nM T17048 C8GA6D 72707984 IC50 = 920 nM T17048 C1Y0VA 73348083 IC50 > 35000 nM T17048 CZHS79 73349449 IC50 = 13800 nM T17048 C7LMU5 73349625 IC50 = 3000 nM T17048 CQB58W 73351007 IC50 = 11200 nM T17048 C38KLY 73351008 IC50 = 16400 nM T17048 C8W4JU 73351009 IC50 = 19700 nM T17048 CWLS07 73351168 IC50 = 3000 nM T17048 CE93QP 73352483 IC50 = 13800 nM T17048 CM08OX 73355679 IC50 = 2000 nM T17048 CW6LC3 73355680 IC50 > 32000 nM T17048 CX49OC 73357045 IC50 = 12000 nM T17048 CV76QL 73357046 IC50 = 9000 nM T17048 CMW35D 73357211 IC50 = 8400 nM T17048 CK40WO 75164138 IC50 > 1000000 nM T17048 CX5CB3 76308343 IC50 = 4500 nM T17048 CG8O6N 76308344 IC50 = 3000 nM T17048 C9WKF4 76308355 IC50 = 19000 nM T17048 C9KJV0 76308356 IC50 = 4100 nM T17048 CQ6FW9 76309460 IC50 = 132 nM T17048 C5Y1VQ 76311989 IC50 = 2900 nM T17048 CN0S3G 76312013 IC50 = 3400 nM T17048 CH2N4W 76312014 IC50 = 16000 nM T17048 CO0T6F 76314922 IC50 > 1000000 nM T17048 CWVY67 76315566 IC50 = 3400 nM T17048 C5ID2K 76315567 IC50 = 4000 nM T17048 C3W2YR 76318541 IC50 = 250000 nM T17048 CE2JA7 76320395 IC50 = 1100 nM T17048 CC5V3E 76320396 IC50 = 592 nM T17048 CU70WJ 76322883 IC50 = 2900 nM T17048 CB80SY 76325813 IC50 = 500000 nM T17048 C9SP5Y 76326426 IC50 = 7100 nM T17048 CKU2E5 76326445 IC50 = 23000 nM T17048 C4XYF0 76326446 IC50 = 2700 nM T17048 CN8UB0 76326447 IC50 = 15000 nM T17048 CUZS03 76326448 IC50 = 350 nM T17048 CNS87J 76329404 IC50 > 1000000 nM T17048 CYJ9X1 76329405 IC50 = 250000 nM T17048 CTV9X8 76330068 IC50 = 20000 nM T17048 C37OGI 76330069 IC50 = 20000 nM T17048 CV9X5P 76331253 IC50 = 3749 nM T17048 C5BW0P 76331254 IC50 = 639 nM T17048 CCEI13 76333693 IC50 = 2100 nM T17048 CWX1I6 76333694 IC50 = 3000 nM T17048 CEK3H5 76333718 IC50 = 12000 nM T17048 C0DK7S 76333719 IC50 = 4000 nM T17048 C9AFJ1 76334830 IC50 = 592 nM T17048 CHG18U 76336671 IC50 = 125000 nM T17048 C3R7DY 88962303 IC50 > 256000 nM T17048 CIKL27 90284582 IC50 > 200000 nM T17048 CQB85S 101233647 IC50 = 176000 nM T17048 CC5H8Q 101233649 IC50 = 64500 nM T17048 CXRV31 102350366 IC50 > 200000 nM T17048 C31SDC 102350368 IC50 = 35200 nM T17048 CMD9E2 110273100 IC50 > 100000 nM T17048 C95LAW 118724649 IC50 = 337000 nM T17048 CD0F4P 122178382 IC50 = 55370 nM T17048 CTZ4B8 122182572 IC50 > 1000000 nM T17048 CG2BL7 122182573 IC50 > 1000000 nM T17048 C4HU8M 122182574 IC50 > 1000000 nM T17048 C4SG2Y 122182575 IC50 > 1000000 nM T17048 CZRS91 122192946 IC50 = 10000 nM T17048 C3L2QW 127024915 IC50 = 900 nM T17048 C93COL 127033765 IC50 = 40000 nM T17048 CJ69CG 127033766 IC50 = 5000 nM T17048 CEH95L 132576588 IC50 = 8100 nM T17048 C7RJ4U 132576589 IC50 = 18500 nM T17048 CC1Z2E 132576591 IC50 = 2430 nM T17048 CKQ9J1 132576592 IC50 = 55300 nM T17048 C0KPG2 132942295 IC50 = 7080 nM T17048 C3PQO4 132942296 IC50 = 5440 nM T17048 CA3M0F 134129981 IC50 > 100000 nM T17048 CR9QA4 134130052 IC50 = 87580 nM T17048 CN0UL5 134130152 IC50 > 100000 nM T17048 C87IXS 134130167 IC50 = 100000 nM T17048 CR35XK 134130204 IC50 = 11250 nM T17048 CIK1X8 134130206 IC50 = 34330 nM T17048 C27NLE 134130331 IC50 = 13900 nM T17048 CFCG09 134130551 IC50 > 100000 nM T17048 C30SMC 134130722 IC50 = 19500 nM T17048 C9GZ8R 134130832 IC50 = 17750 nM T17048 CB45CO 134130860 IC50 > 100000 nM T17048 CXGP69 134130865 IC50 > 100000 nM T17048 CV8A1M 134130889 IC50 = 5140 nM T17048 C7FQO0 134131013 IC50 = 19440 nM T17048 CW96HI 134131206 IC50 > 100000 nM T17048 CDK5S7 134131300 IC50 = 35650 nM T17048 CJ0X4W 134131366 IC50 = 23770 nM T17048 C0SHV2 134131490 IC50 > 100000 nM T17048 C21MIC 134346930 IC50 = 125000 nM T17048 C6UCR1 134346933 IC50 = 1950 nM T17048 C2V9ZE 134346935 IC50 = 1950 nM T17048 CXUN93 134346942 IC50 = 3900 nM T17048 CW3OC5 134346944 IC50 = 15600 nM T17048 C5OQN6 134346949 IC50 = 3900 nM T17048 C57BSY 134589805 IC50 = 164600 nM T17048 C41PKX 134603873 IC50 = 127600 nM T17048 CG4SM8 134816158 IC50 = 970 nM T17048 C0BAY3 135465927 IC50 = 20000 nM T17048 C36GSJ 135611993 IC50 > 1000000 nM T17048 C6ZJX8 135874968 IC50 > 1000000 nM T17048 CQ0KL8 135883794 IC50 > 1000000 nM T17048 CN70KL 135887676 IC50 > 1000000 nM T17048 CLEY16 136110933 IC50 = 34930 nM T17048 CFP0O5 136233034 IC50 = 46500 nM T17048 CGL12X 137631661 IC50 = 10000 nM T17048 CD2U7Z 137636268 IC50 = 13400 nM T17048 C1CID8 137636431 IC50 = 150000 nM T17048 CTV3A5 137636616 IC50 = 99100 nM T17048 CH67OK 137637192 IC50 = 10000 nM T17048 CA29UL 137637498 IC50 = 1000 nM T17048 CNZ10L 137637897 IC50 = 7000 nM T17048 CG02BV 137638495 IC50 < 10000 nM T17048 CU6HD0 137639202 IC50 <= 2500 nM T17048 C6WK4E 137639369 IC50 > 200000 nM T17048 C2SC9H 137640814 IC50 = 10000 nM T17048 C9VL0H 137642577 IC50 = 137000 nM T17048 CVKH90 137643817 IC50 = 16100 nM T17048 CDC16Z 137644529 IC50 = 4880 nM T17048 CH4N3E 137644827 IC50 = 10000 nM T17048 C03VDC 137645384 IC50 = 1500 nM T17048 CK42IG 137646471 IC50 > 100000 nM T17048 C2E1QG 137646796 IC50 = 10000 nM T17048 C9U3XY 137647086 IC50 = 5500 nM T17048 CKIQ30 137647664 IC50 = 89200 nM T17048 CP05EN 137648380 IC50 = 5000 nM T17048 CDO57G 137653088 IC50 = 10000 nM T17048 CD9PF4 137653213 IC50 = 8100 nM T17048 C3P4JU 137653544 IC50 = 52890 nM T17048 CTG1M0 137655122 IC50 = 10000 nM T17048 C7ZYW9 137655794 IC50 = 2200 nM T17048 CTFW15 137656076 IC50 = 29060 nM T17048 CX29KZ 137656647 IC50 = 55700 nM T17048 CWH38X 137661070 IC50 = 2500 nM T17048 CY32GM 137662151 IC50 = 200000 nM T17048 CE8AK6 137662271 IC50 = 120000 nM T17048 CC9K8L 137796790 IC50 = 210000 nM T17048 CT9W7K 145967676 IC50 = 3000 nM T17048 C8K9RX 145969134 IC50 = 26100 nM T17048 CV89SL 145980592 IC50 = 1940 nM T17048 CDO21B 145982399 IC50 = 1190 nM T17048 C6VTY7 145982697 IC50 = 2980 nM T17048 C40OAP 145987091 IC50 = 2970 nM T17048 CY0D3V 145988517 IC50 = 1220 nM T17048 CKB7J0 145990364 IC50 = 5380 nM T17048 CS5WR7 145991174 IC50 = 850 nM T17048 CW6HX8 145992254 IC50 = 940 nM T17048 CV2AE1 145993394 IC50 = 2120 nM T17048 C1TAC4 146499656 IC50 > 200000 nM T17048 C8P3GC 146499745 IC50 > 200000 nM T17048 CXG41R 146538922 IC50 > 200000 nM T17048 CXO50E 146539013 IC50 = 128400 nM T17048 CL86WZ 146539124 IC50 > 200000 nM T17048 C4J2TL 155168924 EC50 = 3100 nM T17048 CL79QN 155186428 EC50 = 3500 nM T17048 CL84NU 155186429 EC50 = 1200 nM T17048 CC8D6T 155186649 EC50 = 1200 nM T17048 CSB28K 155186660 IC50 = 9000 nM T17048 C3K4FP 155186662 EC50 = 1700 nM T17048 CK6VP5 155186665 IC50 = 5000 nM T17048 CM6GB3 155186668 EC50 = 1100 nM T17048 CAG9S1 155510469 IC50 = 3400 nM T17048 CZO2D3 155511481 IC50 = 126600 nM T17048 COX79T 155511733 IC50 > 1000000 nM T17048 C2YH5W 155511964 IC50 = 451400 nM T17048 C2J6ET 155512524 IC50 = 55500 nM T17048 COAS54 155515372 IC50 = 28000 nM T17048 C78SKX 155517816 IC50 = 9200 nM T17048 CALX19 155517971 IC50 = 154900 nM T17048 CW41ZQ 155519351 IC50 = 36700 nM T17048 CGY2H4 155521271 IC50 = 9200 nM T17048 C37LVE 155521285 IC50 = 164100 nM T17048 C6M0IE 155521664 IC50 > 200000 nM T17048 C7R5WZ 155523504 IC50 = 43200 nM T17048 C73JPD 155524074 EC50 = 1000 nM T17048 CX7DJ5 155524997 IC50 = 55300 nM T17048 CI29ED 155525113 IC50 = 8300 nM T17048 CL32BV 155525436 IC50 = 36900 nM T17048 CGH04E 155525473 IC50 = 22500 nM T17048 CRC9T2 155526033 IC50 = 1200 nM T17048 C6YWL3 155527728 IC50 = 10200 nM T17048 C3L8CA 155528225 IC50 = 22500 nM T17048 C8W4TC 155528870 IC50 = 12400 nM T17048 CXK6D9 155529160 IC50 = 54200 nM T17048 CG3H1V 155529474 IC50 = 2000 nM T17048 C0RA1N 155530384 IC50 = 34400 nM T17048 CF3YZ5 155531933 IC50 = 716000 nM T17048 C61ZSK 155532193 IC50 = 8100 nM T17048 CU6V9E 155532517 IC50 = 7800 nM T17048 C60SDZ 155535581 IC50 = 129100 nM T17048 C05VXM 155535908 IC50 = 170800 nM T17048 C0W9RH 155536642 IC50 = 15100 nM T17048 C0Y4PN 155536985 IC50 = 34000 nM T17048 CA4DB0 155537116 IC50 = 293400 nM T17048 C8D3EK 155537498 EC50 = 2400 nM T17048 CUS3N5 155537510 IC50 = 36600 nM T17048 C5Y7UQ 155544885 IC50 = 145100 nM T17048 C2EI0B 155545322 IC50 = 10200 nM T17048 CTNU51 155546705 IC50 = 7300 nM T17048 CQ6D2C 155547369 IC50 > 200000 nM T17048 CJK8H2 155547483 IC50 = 14400 nM T17048 C2AF0E 155548810 IC50 = 38600 nM T17048 C0T1XK 155549458 IC50 = 422100 nM T17048 CSL90Q 155550022 IC50 = 15800 nM T17048 C3C1HN 155550686 IC50 = 84000 nM T17048 C2VH3K 155551829 IC50 = 107800 nM T17048 C7O5MY 155552722 IC50 = 161400 nM T17048 CYU9S2 155553790 IC50 = 11400 nM T17048 C62SYX 155554446 IC50 = 128400 nM T17048 C6BR0V 155554872 IC50 = 11100 nM T17048 CYE87L 155554944 IC50 > 1000000 nM T17048 C0M2SO 155555214 IC50 = 388100 nM T17048 CN0O8I 155555409 IC50 = 700 nM T17048 CZB10X 155558124 IC50 = 268900 nM T17048 CRIQ42 155559615 IC50 = 38700 nM T17048 C52WCD 155562094 IC50 = 9700 nM T17048 CN21FD 155562417 IC50 = 8400 nM T17048 CESW65 155563883 IC50 = 8400 nM T17048 CB5V4E 155567888 IC50 = 45300 nM T17048 C7X4BH 155568248 IC50 = 156600 nM T17048 CJA97M 155568579 IC50 = 165600 nM T17048 C70DMV 155568695 IC50 = 74400 nM T17048 D00DNY 3213 IC50 = 3300 nM T17048 D01BKS 9918693 IC50 > 250000 nM T17048 D02NCW 15601738 IC50 = 17500 nM T17048 D05KJY 72326 IC50 = 38600 nM T17048 D0E8ZH 2392 IC50 = 28920 nM T17048 D0HD2G 4788 IC50 = 46.1 ug.mL-1 T17048 D0I0HL 10391130 IC50 = 17600 nM T17048 D0L8BN 44559995 IC50 = 4000 nM T17048 D0MF5Y 5281614 IC50 = 8.2 ug.mL-1 T17048 D0NJ4H 5281670 IC50 = 40.8 ug.mL-1 T17048 D0RA6H 259846 IC50 = 10400 nM T17048 D0T3PW 5281672 IC50 = 11.9 ug.mL-1 T57654 D08DHN 67286591 EC50 = 0.6 nM T57654 CF18BX 135217926 EC50 = 0.06 nM T57654 CQ8YW3 142462986 EC50 = 12 nM T57654 C5MDP4 145401914 EC50 = 14 nM T57654 CLK24V 145401954 EC50 = 0.5 nM T57654 C5T6DI 145401976 EC50 = 0.2 nM T57654 C4B3IQ 145401999 EC50 = 5.3 nM T57654 C87IZY 145402050 EC50 = 5.5 nM T57654 C8B7GP 153694344 EC50 = 230 nM T57654 COH19K 155280053 EC50 = 220 nM T57654 CXR1N4 155510680 EC50 = 0.5 nM T57654 CQSY80 155511697 EC50 = 3 nM T57654 CVN93K 155517311 EC50 = 4 nM T57654 C0G4VQ 155527252 EC50 = 9.6 nM T57654 CR84VW 155530488 EC50 = 20 nM T57654 C6ULP5 155533598 EC50 = 2.6 nM T57654 C0UXM5 155534281 EC50 = 2.8 nM T57654 CFHE71 155535392 EC50 = 0.2 nM T57654 CG62IA 155538538 EC50 = 10 nM T57654 CP9Y3F 155542018 EC50 = 2000 nM T57654 CF3R2H 155543036 EC50 = 11 nM T57654 CVG17B 155543929 EC50 = 10 nM T57654 C76WAH 155544352 EC50 = 12 nM T57654 C2MY6S 155544800 EC50 = 13 nM T57654 CUA5M7 155545666 EC50 = 4.5 nM T57654 C01ZOS 155545801 EC50 = 11 nM T57654 C51HXU 155548819 EC50 = 110 nM T57654 C4NQ7Y 155549152 EC50 = 450 nM T57654 C7TKF8 155551474 EC50 = 24 nM T57654 C38VBK 155553283 EC50 = 1.4 nM T57654 C4CWO9 155562598 EC50 = 0.4 nM T57654 CV3H1S 155565183 EC50 = 70 nM T57654 CWM54Q 155568031 EC50 = 190 nM T67231 CA28RG 44433025 IC50 = 1400 nM T67231 CSI19H 44433026 IC50 = 9000 nM T67231 CARE56 44433027 IC50 = 9600 nM T67231 C0NH1E 44433028 IC50 = 540 nM T67231 C9Z6UK 44433029 IC50 = 310 nM T67231 CPJI05 44433030 IC50 = 840 nM T67231 CQ39AW 44433031 IC50 = 590 nM T67231 C5TOX4 44433032 IC50 > 5000 nM T67231 C4FLY7 44433033 IC50 = 430 nM T67231 CK48CX 44433034 IC50 = 3700 nM T67231 CER76A 44433035 IC50 = 510 nM T67231 CN73XZ 44433036 IC50 = 1600 nM T67231 CYJ14E 44433037 IC50 > 16000 nM T67231 C4IS8L 44433038 IC50 > 30000 nM T67231 CIO63X 44433039 IC50 > 30000 nM T67231 CTY6N1 44433040 IC50 > 30000 nM T67231 CG7VX4 44433041 IC50 > 30000 nM T67231 CKP25V 44433042 IC50 > 30000 nM T67231 C4EM1H 44433043 IC50 > 30000 nM T67231 C2QT0W 44433045 IC50 = 37 nM T67231 CK8M5S 44433047 IC50 = 8 nM T67231 C3IU1H 44433049 IC50 = 29 nM T67231 CY5U6X 44433050 IC50 = 95 nM T67231 CC54QY 44433051 IC50 = 100 nM T67231 CO78PY 44433052 IC50 = 250 nM T67231 CK4HC1 44433053 IC50 = 140 nM T67231 C57SJZ 44433054 IC50 = 160 nM T67231 CM1F6Q 44433055 IC50 = 970 nM T67231 CQ64LH 49798318 Ki = 125000 nM T67231 CG6H9M 49798319 Ki = 11800 nM T67231 CEP3Q0 49798321 Ki = 75000 nM T67231 C5URL1 49798322 Ki = 225000 nM T67231 CG2W1O 49798344 Ki = 265000 nM T67231 C8R5EY 49798345 Ki = 140000 nM T67231 D0P7NY 23661637 IC50 = 170 nM T39677 CN67CR 555078 IC50 = 11000 nM T39677 C8XNE3 10198662 Ki = 25 nM T39677 CD4B1N 10488207 Ki = 40 nM T39677 CG71MW 10705248 Ki = 58 nM T39677 CX7KA0 10729666 Ki = 60 nM T39677 CQ96CB 10774930 Ki = 2300 nM T39677 C3RV7P 10778354 Ki = 580 nM T39677 C5IXD3 10823157 Ki = 2200 nM T39677 CUC8N5 25141405 IC50 > 100000 nM T39677 CIT5G7 44561891 IC50 > 100000 nM T39677 C90BGR 44561892 IC50 > 100000 nM T39677 C9RGX4 44561893 IC50 > 100000 nM T39677 CU7NP5 44561930 IC50 > 100000 nM T39677 CV21IQ 44561931 IC50 > 100000 nM T39677 CR08WA 44561932 IC50 > 100000 nM T39677 CJH50R 49797481 IC50 > 100000 nM T54644 D02AIN 122678117 IC50 > 32000 nM T54644 D04TNT 46851313 IC50 = 2300 nM T54644 D0F4GF 24765479 IC50 = 8.2 nM T54644 D0W8XT 60663 IC50 = 32 nM T54644 D0IU2F 4988454 IC50 = 45000 nM T54644 CMT3P0 480764 IC50 = 1000 nM T54644 C1AQ4G 2870439 IC50 = 5390 nM T54644 CUQ4R7 2987239 IC50 > 10000 nM T54644 C0F8EP 3519901 IC50 = 1000 nM T54644 C8KN4J 3876755 IC50 = 68 nM T54644 CZ8TQ5 3944785 IC50 = 281 nM T54644 CVBA68 4101623 IC50 = 5000 nM T54644 CRCD67 4200092 IC50 = 3000 nM T54644 CNZ1F7 6458316 IC50 > 10000 nM T54644 CP5NF6 6461757 IC50 = 610 nM T54644 CJO8N6 10117450 IC50 = 149 nM T54644 CCV0U6 11444582 IC50 = 110 nM T54644 CKB41R 11497976 IC50 = 1700 nM T54644 C3APF9 11563321 IC50 = 420 nM T54644 CKI38O 11684953 IC50 = 540 nM T54644 C9ITW7 11692799 IC50 = 240 nM T54644 CD34SB 15982534 IC50 > 333000 nM T54644 CR7XF5 22084904 IC50 = 2000 nM T54644 C90CGS 24829433 IC50 = 340 nM T54644 CS40MV 24829434 IC50 = 177 nM T54644 C5V9KB 24831706 IC50 = 214 nM T54644 CRB28T 24831868 IC50 = 138 nM T54644 C4RJ2E 24898117 IC50 = 398 nM T54644 CDO93A 24898118 IC50 = 410 nM T54644 CI52SD 24898332 IC50 = 256 nM T54644 CH5JR1 24936279 IC50 = 71 nM T54644 C97EIS 24936281 IC50 = 44 nM T54644 CO98VJ 24938185 IC50 = 29 nM T54644 COT4J1 24954146 IC50 = 2258 nM T54644 CK0QG9 24954512 IC50 = 1251 nM T54644 C0HW1M 24955598 IC50 = 390 nM T54644 C1REU6 35537998 IC50 = 280 nM T54644 C5L9MY 39779000 IC50 = 1000 nM T54644 CL92PJ 44455579 IC50 = 180 nM T54644 C1ATC9 46203893 IC50 = 217 nM T54644 CHTV13 46203894 IC50 = 184 nM T54644 CFYP54 46203897 IC50 = 84 nM T54644 C9L4KT 46205341 IC50 > 333000 nM T54644 CL41FE 46206000 IC50 > 100000 nM T54644 CJW0P1 46852596 IC50 = 19000 nM T54644 CRP91J 46853381 IC50 = 10600 nM T54644 C7K0QO 49862856 IC50 = 139 nM T54644 C0VQ9A 49862857 IC50 = 351 nM T54644 CG62QB 49862858 IC50 = 224 nM T54644 CD4I8G 49862859 IC50 = 247 nM T54644 C73HEN 49862885 IC50 = 104 nM T54644 C9ZO1B 49862925 IC50 = 410 nM T54644 C1SG3L 49862926 IC50 = 800 nM T54644 C5WY7S 49862927 IC50 = 920 nM T54644 C0C7GF 49862958 IC50 = 172 nM T54644 C5XA6G 49862992 IC50 = 146 nM T54644 CH3K1V 49862993 IC50 = 109 nM T54644 CQ06YU 49863039 IC50 = 45 nM T54644 C78JIQ 49863040 IC50 = 182 nM T54644 CJNP67 49863041 IC50 = 251 nM T54644 C95PUV 49863084 IC50 = 3333 nM T54644 CZN36V 49863085 IC50 = 82 nM T54644 CZP63E 49863086 IC50 = 3200 nM T54644 CON50R 49863110 IC50 = 1060 nM T54644 CP94IE 49863137 IC50 = 41 nM T54644 C19RFZ 49863138 IC50 = 176 nM T54644 C1M5LN 49863173 IC50 = 41 nM T54644 C83ECF 49863174 IC50 = 17 nM T54644 C1JIG3 49863206 IC50 = 116 nM T54644 C3XC4A 49863207 IC50 = 57 nM T54644 CL2E5I 49863241 IC50 = 200 nM T54644 CSVC02 49863242 IC50 = 698 nM T54644 CPR56Y 49863257 IC50 = 519 nM T54644 C5EXM2 49863274 IC50 = 84 nM T54644 C04BHX 49863311 IC50 = 35 nM T54644 CWN9I1 49863312 IC50 = 325 nM T54644 C4BHF8 49863313 IC50 = 827 nM T54644 CUDE92 50898773 IC50 = 3600 nM T54644 CPS12B 53317097 IC50 = 92 nM T54644 C2D3HQ 60168069 IC50 > 100000 nM T54644 CL1RV4 67447319 IC50 = 398 nM T54644 CJ7FG0 67448236 IC50 = 350 nM T54644 CC9S6H 67449145 IC50 = 224 nM T54644 COP01E 71517044 IC50 = 2400 nM T54644 C95BFG 71517045 IC50 = 900 nM T54644 C1N2HF 71517046 IC50 = 300 nM T54644 C7GS4P 71517047 IC50 = 500 nM T54644 CWLO57 71517048 IC50 = 500 nM T54644 C87CZW 71517049 IC50 = 3300 nM T54644 CY0VJ8 71517192 IC50 = 400 nM T54644 C5S0XY 71517194 IC50 = 800 nM T54644 C31DLT 71517195 IC50 = 500 nM T54644 CRG0P7 71517196 IC50 = 600 nM T54644 CA07TC 71517197 IC50 = 600 nM T54644 CQKA86 71519342 IC50 = 4900 nM T54644 C2JFW9 71519494 IC50 = 3000 nM T54644 CIG9W3 71519495 IC50 = 1300 nM T54644 CZ03XO 71519496 IC50 = 500 nM T54644 CU71MB 71519497 IC50 = 1200 nM T54644 CBKY29 71519498 IC50 = 1200 nM T54644 CO7B8C 71720776 IC50 = 800 nM T54644 CLXH36 72793718 IC50 = 5800 nM T54644 C3Q1PF 75094570 IC50 = 310 nM T54644 CF7GZ5 86292750 IC50 = 2500 nM T54644 CF7Y2I 86292753 IC50 = 8200 nM T54644 CV8OI5 86292754 IC50 = 10790 nM T54644 CDV37Y 86292938 IC50 = 2890 nM T54644 CEJK10 92135927 IC50 = 5800 nM T54644 CG60JW 117700665 IC50 = 8870 nM T54644 C9YU5M 118512798 IC50 = 4300 nM T54644 C48PFK 118512802 IC50 = 2080 nM T54644 CLHP58 118560158 IC50 = 12 nM T54644 C9S4YL 118560191 IC50 = 14 nM T54644 C0LR9M 118560290 IC50 = 7.8 nM T54644 C7Y8FJ 118560322 IC50 = 10 nM T54644 CE6O4V 118560356 IC50 = 20 nM T54644 CMAN70 118560393 IC50 = 46 nM T54644 C4VG3F 118560394 IC50 = 10 nM T54644 CZ6O0E 118560399 IC50 = 5.1 nM T54644 CVRO18 118560401 IC50 = 4.1 nM T54644 CZ62GY 118560409 IC50 = 3.4 nM T54644 CL12OZ 118560423 IC50 = 21 nM T54644 CH84UX 118560458 IC50 = 13 nM T54644 C7Y2LQ 118560466 IC50 = 220 nM T54644 C0JAX6 118560472 IC50 = 47 nM T54644 CDJL48 118560488 IC50 = 5.3 nM T54644 CY2KI3 118560543 IC50 = 32 nM T54644 C37PDX 118560579 IC50 = 35 nM T54644 CG25JS 118560588 IC50 = 14 nM T54644 CLK32A 118560592 IC50 = 6 nM T54644 C04FRX 118560613 IC50 = 11 nM T54644 CB41MH 118560618 IC50 = 18 nM T54644 CS0RQ3 118560699 IC50 = 7.5 nM T54644 CQG3K7 118560709 IC50 = 6.1 nM T54644 C2DA9Z 118962193 IC50 = 8.6 nM T54644 CHD26A 121596332 IC50 > 33300 nM T54644 C7KNL3 122187207 IC50 = 318 nM T54644 CYE4O0 122187208 IC50 = 132 nM T54644 C8Y5VF 122187209 IC50 = 113 nM T54644 CJ5OR3 122187210 IC50 = 107 nM T54644 CR5TW0 122187211 IC50 = 76 nM T54644 CA89DJ 122187212 IC50 = 361 nM T54644 CR2Q6E 122187213 IC50 = 210 nM T54644 CA3K1Y 122187853 IC50 = 2065 nM T54644 CI1NX6 122187854 IC50 = 207 nM T54644 C91RFU 122187855 IC50 = 193 nM T54644 CN7I3U 122187856 IC50 = 557 nM T54644 C1YK2E 122678192 IC50 > 32000 nM T54644 CF6D2P 126740597 IC50 = 6.7 nM T54644 CAYS28 126740598 IC50 = 140 nM T54644 CIQ23U 126740608 IC50 = 7.8 nM T54644 C1O5VB 126740610 IC50 = 25 nM T54644 C9KEY6 126740618 IC50 = 18 nM T54644 CA1M2Q 126740623 IC50 = 8.4 nM T54644 CNUF36 126740624 IC50 = 3.8 nM T54644 COE64S 126740626 IC50 = 7 nM T54644 CS2Y3W 126740650 IC50 = 15 nM T54644 CHO17P 126740652 IC50 = 4.3 nM T54644 CKNV98 126740697 IC50 = 34 nM T54644 CJR57G 132609277 IC50 = 2520 nM T54644 CRAG89 132609278 IC50 = 2320 nM T54644 CM4U6T 132961366 IC50 = 340 nM T54644 C0AI1V 132991411 IC50 = 102 nM T54644 C1XR9I 134130259 IC50 = 241 nM T54644 C3P7TZ 134130807 IC50 = 61 nM T54644 C9RZB3 134131854 IC50 = 205 nM T54644 CW0Q7I 134132801 IC50 = 55 nM T54644 CS0A8O 134132803 IC50 = 330 nM T54644 C58IKL 134133106 IC50 = 900 nM T54644 CHR09A 134133339 IC50 = 240 nM T54644 C40FOB 134133525 IC50 = 140 nM T54644 CG21YN 134133529 IC50 = 682 nM T54644 CE32KO 134133599 IC50 = 28 nM T54644 CH9MI7 134133901 IC50 = 414 nM T54644 C3GIH1 134134030 IC50 = 31 nM T54644 CEWV89 134134318 IC50 = 14 nM T54644 C5RY7Q 134134580 IC50 = 61 nM T54644 CS6Z7U 134135105 IC50 = 430 nM T54644 CBC5I3 134135133 IC50 = 198 nM T54644 C67QGZ 134135164 IC50 = 9 nM T54644 CV0I4O 134135871 IC50 = 6 nM T54644 CJM8S0 134135899 IC50 = 30 nM T54644 CQ54CZ 134135912 IC50 = 231 nM T54644 CMQV20 134136121 IC50 > 10000 nM T54644 C4SB8F 134136300 IC50 = 690 nM T54644 CK9MG1 134136380 IC50 = 33 nM T54644 C5VG6N 134136586 IC50 = 16 nM T54644 C3W6FX 134137496 IC50 = 110 nM T54644 CW5T6X 134138179 IC50 = 420 nM T54644 CJ4T0C 134138248 IC50 > 11550 nM T54644 CW4BU5 134138250 IC50 = 93 nM T54644 CLW07U 134138308 IC50 = 72 nM T54644 CERI05 134138759 IC50 = 14 nM T54644 CSEW05 134139055 IC50 = 240 nM T54644 CAFS70 134139103 IC50 = 447 nM T54644 C07AWK 134139327 IC50 = 410 nM T54644 C29IBJ 134139406 IC50 = 815 nM T54644 CPG8R2 134139460 IC50 > 8580 nM T54644 CRJ72V 134140275 IC50 = 25 nM T54644 C9CO2P 134140278 IC50 = 66 nM T54644 CQ6V1Z 134140414 IC50 = 320 nM T54644 C39PGW 134140468 IC50 = 1490 nM T54644 CWI1J7 134140478 IC50 = 14600 nM T54644 C9IMS2 134140658 IC50 = 382 nM T54644 C8L5VZ 134140864 IC50 = 11 nM T54644 C62AVQ 134141003 IC50 = 59 nM T54644 C3NRL2 134141387 IC50 = 44 nM T54644 CZ06DO 134141633 IC50 = 33 nM T54644 CIPG12 134141754 IC50 > 6400 nM T54644 C90WMC 134141766 IC50 = 530 nM T54644 CR29YW 134141773 IC50 = 95 nM T54644 C4IV9M 134141806 IC50 > 6500 nM T54644 CGA34U 134141893 IC50 = 604 nM T54644 C6U2PJ 134142122 IC50 = 52 nM T54644 C0CT2A 134142164 IC50 = 62 nM T54644 C4KI8G 134142247 IC50 = 613 nM T54644 CVC5M6 134142399 IC50 = 860 nM T54644 CXK8D7 134142518 IC50 = 15 nM T54644 C16TWR 134142614 IC50 = 305 nM T54644 C2VSP7 134143155 IC50 = 62 nM T54644 CQ80GN 134143440 IC50 = 112 nM T54644 C1PT9H 134143519 IC50 = 17 nM T54644 CEG7S4 134143554 IC50 = 36 nM T54644 CH03BE 134143575 IC50 = 104 nM T54644 C2VJ7N 134143801 IC50 > 7300 nM T54644 C9A1XL 134143901 IC50 > 11000 nM T54644 CS7G2P 134144179 IC50 = 48 nM T54644 C1OLQ9 134144496 IC50 = 358 nM T54644 C8XR0U 134145066 IC50 = 225 nM T54644 CTIX18 134145629 IC50 = 350 nM T54644 CN8WV9 134145759 IC50 = 31 nM T54644 C6OD8Y 134145781 IC50 = 22 nM T54644 CB6QF0 134145994 IC50 = 38 nM T54644 C7GL6O 134146020 IC50 = 72 nM T54644 CY5ME7 134146171 IC50 = 33 nM T54644 CT0KP6 134146400 IC50 = 316 nM T54644 CG7RX1 134146440 IC50 = 860 nM T54644 CN2ST6 134146817 IC50 > 10700 nM T54644 CE15VD 134146997 IC50 = 42 nM T54644 CV73DS 134147142 IC50 = 835 nM T54644 CU0WK1 134147287 IC50 = 2670 nM T54644 C1JXF2 134147318 IC50 = 55 nM T54644 C6J0RP 134147643 IC50 = 1600 nM T54644 CHN1C9 134147829 IC50 = 9010 nM T54644 C0ZQM8 134147890 IC50 = 500 nM T54644 CHF36J 134147928 IC50 = 70 nM T54644 C5C7BZ 134147980 IC50 = 922 nM T54644 C1WSQ6 134148112 IC50 = 120 nM T54644 C9W1AN 134148285 IC50 = 464 nM T54644 CW9M8G 134148369 IC50 = 44 nM T54644 C45XMS 134148468 IC50 = 14 nM T54644 C20MDR 134148760 IC50 = 68 nM T54644 C36CTV 134149105 IC50 > 5300 nM T54644 CWZ47K 134149196 IC50 = 24 nM T54644 CRBG97 134149384 IC50 = 420 nM T54644 C1UY6K 134149672 IC50 = 12 nM T54644 CYQ43A 134149751 IC50 = 841 nM T54644 C4FC6U 134149941 IC50 = 18 nM T54644 CJZ29K 134149992 IC50 > 11000 nM T54644 CM9ZY1 134150199 IC50 = 46 nM T54644 CJQ37D 134150323 IC50 = 393 nM T54644 CI58UE 134150489 IC50 = 55 nM T54644 CW38EV 134150541 IC50 = 40 nM T54644 CML57E 134151608 IC50 = 49 nM T54644 CO1JA4 134151710 IC50 = 340 nM T54644 CV25WH 134151973 IC50 = 479 nM T54644 C0NU4T 134152220 IC50 = 47 nM T54644 CVLO27 134152587 IC50 = 58 nM T54644 CPB68S 134152614 IC50 = 21 nM T54644 C7TV2H 134152703 IC50 = 212 nM T54644 CKI47N 134152745 IC50 = 392 nM T54644 C7NV2W 134152994 IC50 = 91 nM T54644 CFK81J 134153093 IC50 = 618 nM T54644 C19LMT 134153241 IC50 = 42 nM T54644 CZX13T 134153284 IC50 = 209 nM T54644 CV9ME7 134153508 IC50 = 13 nM T54644 C4L8QS 134153676 IC50 = 7410 nM T54644 C0V6YF 134153738 IC50 = 95 nM T54644 CEA6H8 134153757 IC50 = 428 nM T54644 CI61JC 134153846 IC50 = 410 nM T54644 CFX72G 134154056 IC50 = 60 nM T54644 CMH28S 134154353 IC50 = 790 nM T54644 C3AW2M 134155076 IC50 = 695 nM T54644 CX8P0D 134155552 IC50 = 141 nM T54644 CUH82M 134155661 IC50 = 202 nM T54644 CN98ZC 134156036 IC50 = 4695 nM T54644 CAS9U3 134156465 IC50 = 224 nM T54644 CE8V5G 134156616 IC50 = 230 nM T54644 C81DUY 134156667 IC50 > 10000 nM T54644 C3O9IA 134156846 IC50 = 25 nM T54644 C9F3EG 134156994 IC50 = 51 nM T54644 CS4PX9 134157075 IC50 > 8000 nM T54644 C5TC7R 134157194 IC50 = 52 nM T54644 CLMT10 134157774 IC50 = 91 nM T54644 CT53LX 137636153 IC50 = 5600 nM T54644 CQ0B2Y 137645508 IC50 = 3390 nM T54644 CV0J6S 137650114 IC50 = 3690 nM T54644 CDS56O 137652520 IC50 = 5100 nM T54644 C05KZL 141634203 IC50 = 120 nM T54644 CJXN76 142550274 IC50 = 260 nM T54644 CXO29N 142550275 IC50 = 500 nM T54644 CE9D2F 142550277 IC50 = 480 nM T54644 CIDN98 142550281 IC50 = 390 nM T54644 CDRF75 142550292 IC50 = 640 nM T54644 C57STC 142550294 IC50 = 460 nM T54644 CM6X2H 142550296 IC50 = 1020 nM T54644 C8CN6R 142550302 IC50 = 1250 nM T54644 CN9O6Q 145963763 IC50 = 21 nM T54644 CBC6A4 145964052 IC50 = 160 nM T54644 CZFE02 145964073 IC50 = 62 nM T54644 C6WB0E 145964120 IC50 = 410 nM T54644 C1RJ5L 145964213 IC50 = 21 nM T54644 C7TAQ5 145964444 IC50 > 10000 nM T54644 CL3J5T 145964488 IC50 = 170 nM T54644 CX7TC4 145964712 IC50 = 160 nM T54644 C0JGD5 145964736 IC50 = 300 nM T54644 CUQD06 145964872 IC50 = 1300 nM T54644 C6V5PA 145965039 IC50 = 370 nM T54644 CSJV78 145965046 IC50 = 750 nM T54644 CEK7F5 145965051 IC50 = 600 nM T54644 CU79FE 145965065 IC50 = 210 nM T54644 C3XZ9G 145965167 IC50 = 57 nM T54644 CZ7VP8 145965333 IC50 = 100 nM T54644 COA0D4 145965395 IC50 = 330 nM T54644 CG5D0A 145965520 IC50 = 23 nM T54644 C2SV8D 145965539 IC50 = 1000 nM T54644 CB24MN 145965576 IC50 = 39 nM T54644 C8MUI9 145965686 IC50 = 27 nM T54644 CM0C4Q 145965785 IC50 = 21 nM T54644 C74GDJ 145965861 IC50 = 280 nM T54644 CSR0W9 145965878 IC50 = 240 nM T54644 CP9GX0 145965960 IC50 = 580 nM T54644 CC25LD 145966135 IC50 = 71 nM T54644 CY6NH0 145966175 IC50 = 110 nM T54644 C6P5GM 145966272 IC50 = 310 nM T54644 C7MOG0 145966280 IC50 = 260 nM T54644 CNG80S 145966315 IC50 = 6300 nM T54644 C3I5WD 145966882 IC50 = 33 nM T54644 CB6G2J 145966887 IC50 = 890 nM T54644 C9OZ7B 145966987 IC50 > 10000 nM T54644 CQ6S4I 145967128 IC50 = 39 nM T54644 CIFN68 145967321 IC50 = 44 nM T54644 C3P6KV 145967526 IC50 = 30 nM T54644 CGV18I 145967628 IC50 = 239000 nM T54644 CQ74PV 145967661 IC50 = 41000 nM T54644 CWRS54 145967754 IC50 = 1450 nM T54644 C7Y0MU 145967892 IC50 = 492000 nM T54644 CE3GA1 145968071 IC50 = 95000 nM T54644 C9GYA8 145968219 IC50 = 600 nM T54644 C5YK7S 145968281 IC50 = 771000 nM T54644 C09HME 145968567 IC50 = 288000 nM T54644 C53KZP 145968632 IC50 = 112000 nM T54644 CM06JK 145968873 IC50 = 110000 nM T54644 C3F9UM 145968918 IC50 = 410 nM T54644 CO1FC6 145968951 IC50 = 5000 nM T54644 C8A3JX 145968953 IC50 = 23 nM T54644 CTE5M6 145968992 IC50 = 270000 nM T54644 C0RFY3 145969009 IC50 = 166000 nM T54644 C7KCA4 145969044 IC50 = 54000 nM T54644 CX2Q3S 145969169 IC50 = 27 nM T54644 CFV2D8 145969191 IC50 = 300000 nM T54644 C3PN7K 145969264 IC50 = 328000 nM T54644 CJ4BF6 145969488 IC50 = 332000 nM T54644 CG56AM 145969886 IC50 = 319000 nM T54644 C9SQV7 145969924 IC50 = 248000 nM T54644 CKX32N 145970126 IC50 = 195000 nM T54644 CXNE63 145970149 IC50 = 153000 nM T54644 C4XD2J 145970156 IC50 = 212000 nM T54644 C3AR7T 145970259 IC50 = 688000 nM T54644 C93RXD 145970771 IC50 > 10000 nM T54644 C0V7HM 145970794 IC50 = 171000 nM T54644 CD9SA3 145970877 IC50 > 1000000 nM T54644 CL9ZA4 145971033 IC50 = 165000 nM T54644 CLQ74T 145971053 IC50 = 521000 nM T54644 C5LCQ7 145971063 IC50 = 498000 nM T54644 CE9P1Z 145971143 IC50 = 64000 nM T54644 CJE56F 145971412 IC50 = 22 nM T54644 CXMQ72 145971782 IC50 = 1100 nM T54644 CM92KQ 145971885 IC50 = 25 nM T54644 CK06VY 145972088 IC50 = 64 nM T54644 CO0FR7 145972093 IC50 = 380 nM T54644 CAOS28 145973012 IC50 = 21 nM T54644 C2C1ST 145973030 IC50 = 55 nM T54644 CQYB38 145973089 IC50 = 38 nM T54644 C8UN1L 145973107 IC50 = 470 nM T54644 C8RFM3 145973261 IC50 > 33000 nM T54644 C2L7RP 145973300 IC50 = 510 nM T54644 CQ7WG9 145973409 IC50 = 20 nM T54644 C1N4UG 145973443 IC50 = 370 nM T54644 CHZ21U 145973703 IC50 = 220 nM T54644 CH9P2S 145973704 IC50 = 3400 nM T54644 CHQ32U 145973751 IC50 = 42 nM T54644 C5OX8I 145973789 IC50 = 90 nM T54644 CON93L 145973912 IC50 = 155 nM T54644 CM78OR 145974461 IC50 = 850 nM T54644 C7B2VG 145974480 IC50 = 2100 nM T54644 C8G1KM 145974485 IC50 = 38 nM T54644 CED15B 145974511 IC50 = 190 nM T54644 C2OL7I 145975061 IC50 = 530 nM T54644 C9UVC6 145975140 IC50 = 5.5 nM T54644 CDB4P8 145975231 IC50 = 990 nM T54644 CR2N8T 145975397 IC50 = 30 nM T54644 C58WOB 145975751 IC50 = 21 nM T54644 C3W2OE 145975832 IC50 = 2150 nM T54644 CMWY20 145975926 IC50 = 1500 nM T54644 C1YSW7 145976102 IC50 = 25 nM T54644 CK8X4G 145976223 IC50 = 56 nM T54644 CO8KN3 145976268 IC50 = 380 nM T54644 CN72ZM 145976351 IC50 > 10000 nM T54644 C4KF1L 145976387 IC50 = 65 nM T54644 C3XE5S 145976394 IC50 = 140 nM T54644 CE50WI 145976410 IC50 = 340 nM T54644 CGA1B5 145976660 IC50 = 370 nM T54644 C2BVH9 145976792 IC50 = 330 nM T54644 C1QU0T 145976799 IC50 = 110 nM T54644 CM6ZT8 145976855 IC50 = 100 nM T54644 CLCM81 145976857 IC50 = 12 nM T54644 C1L2NM 145977186 IC50 = 1040 nM T54644 C0S3TG 145977189 IC50 = 1900 nM T54644 CH3FM6 145977296 IC50 = 74 nM T54644 CAR4F9 145977337 IC50 = 590 nM T54644 C5I6VA 145977340 IC50 = 21 nM T54644 C21VED 145977676 IC50 = 670 nM T54644 CU38DI 145977733 IC50 = 400 nM T54644 CSE52C 145977745 IC50 = 61 nM T54644 C45HOF 145977787 IC50 = 10 nM T54644 C1XD8F 145977860 IC50 = 160 nM T54644 CCL06J 145977910 IC50 = 350 nM T54644 CI89TQ 145978258 IC50 = 290 nM T54644 C8BD3R 145978287 IC50 = 820 nM T54644 C7DV6A 145978317 IC50 = 31 nM T54644 CL36DE 145978466 IC50 = 210 nM T54644 CU0N4O 145978657 IC50 = 36 nM T54644 CGW6Q5 145978668 IC50 = 6.6 nM T54644 C98BZP 145986355 IC50 = 109000 nM T54644 C4NP8S 145988617 IC50 > 1000000 nM T54644 CA2XP0 145988629 IC50 = 326000 nM T54644 CV4LT9 153635960 IC50 = 7610 nM T54644 D0T6NE 44540045 IC50 = 73 nM T54644 D0VE0Q 72936 IC50 = 1000 nM T92521 D00ZFP 5870 IC50 > 50000 nM T92521 D02YIZ 12560 IC50 = 40000 nM T92521 D04AIT 5280445 Ki = 56 nM T92521 D06XMU 6013 Ki = 411800 nM T92521 D07MGA 72281 IC50 = 511 nM T92521 D08QMX 5757 Ki = 1900 nM T92521 D0AN7B 896 Ki = 14000 nM T92521 D0G4KG 3828 IC50 = 34600 nM T92521 D0K8KX 5280343 Ki = 23 nM T92521 D0TR5X 3386 IC50 = 475000 nM T92521 D0W8WB 2353 Ki = 44 nM T92521 D06NYA 66414 Ki = 36000 nM T92521 D0G5CS 68071 IC50 = 1679 nM T92521 D0H9YO 133967 IC50 = 500 nM T92521 D0QR5G 2355 IC50 = 15300 nM T92521 D0U3EP 445154 Ki = 750 nM T92521 D02NYK 9929138 Ki = 4.38 nM T92521 D0S2HO 10819 Ki = 2000 nM T92521 C6X9CB 978 IC50 > 120000 nM T92521 CQ4X7V 3433 Ki > 200000 nM T92521 CM1G6U 5708 IC50 = 130 nM T92521 CMOP10 5889 IC50 = 9 nM T92521 CK4N7S 6293 Ki = 500 nM T92521 CWH70F 31423 IC50 = 2 nM T92521 COZX93 61322 Ki = 7460 nM T92521 CY5KZ7 63090 IC50 = 11 nM T92521 CPW9B5 65752 IC50 = 55 nM T92521 CMLI08 68079 IC50 = 6380 nM T92521 C09AHX 68081 Ki = 6000 nM T92521 CL9WU4 68578 Ki = 149000 nM T92521 CL7D5O 97214 Ki = 35 nM T92521 CL97OF 97548 IC50 = 7.3 nM T92521 CZB67X 98608 IC50 = 220 nM T92521 CZX39C 101450 IC50 = 130 nM T92521 C14HXK 148756 IC50 = 55 nM T92521 CM2H7V 152430 IC50 = 2500 nM T92521 C4VCM7 156372 IC50 = 330 nM T92521 CQ6E7B 160237 Ki > 800 nM T92521 C1R6GB 189060 IC50 = 7700 nM T92521 C2C4VM 280475 IC50 = 2000 nM T92521 CVD3L1 282535 IC50 = 163000 nM T92521 CIS4M5 363209 IC50 = 9900 nM T92521 C1DQV0 378227 IC50 = 84 nM T92521 CS34TJ 378228 IC50 = 110 nM T92521 C7HME8 439246 IC50 = 3656 nM T92521 CVH49X 480768 EC50 = 5200 nM T92521 C3RT9P 676300 IC50 = 43.4 nM T92521 C2YJ8D 688838 IC50 = 14.8 nM T92521 C2AHB4 689051 IC50 = 6040 nM T92521 CY1BQ5 799928 IC50 = 400000 nM T92521 CP2DH7 830498 IC50 = 57 nM T92521 C2WP5U 3084288 IC50 = 4100 nM T92521 CBO10S 3419544 IC50 = 7000 nM T92521 CQX12K 5197944 IC50 = 5.1 nM T92521 C8ELV4 5281617 Ki > 2340 nM T92521 CK5NZ0 5319487 IC50 = 71 nM T92521 COJI90 5338258 IC50 = 650 nM T92521 CWFP51 5338324 IC50 = 2110 nM T92521 CI6TE3 5348770 IC50 = 157.7 nM T92521 C5E9XW 5351234 IC50 = 19 nM T92521 CK7WJ9 5354004 IC50 = 2 nM T92521 C5Z0HQ 5355549 IC50 = 77 nM T92521 C51QVL 5355551 IC50 = 95.5 nM T92521 C4G5QC 5387294 IC50 = 3000 nM T92521 CZ1U8A 5468167 IC50 = 176 nM T92521 CUL7A5 5471349 Ki = 587000 nM T92521 CLX57S 5473050 Ki = 900 nM T92521 CBPK50 5717022 IC50 = 525 nM T92521 CPT10H 5717399 IC50 = 29 nM T92521 C21EJH 5717404 IC50 = 19 nM T92521 CE9KZ5 5720628 IC50 = 93 nM T92521 CH16ZG 5729125 IC50 = 40.2 nM T92521 CJMQ48 5737900 IC50 = 13000 nM T92521 CSH9C1 5787676 IC50 > 20000 nM T92521 CMWC08 5837372 EC50 = 10000 nM T92521 CAJK62 5859537 IC50 = 5200 nM T92521 CNL31B 5920936 IC50 = 37.8 nM T92521 CBM02K 5926900 IC50 = 349 nM T92521 CX23PO 6020016 IC50 = 200 nM T92521 CZ5N4R 6020915 IC50 = 466 nM T92521 C2V8QP 6174007 IC50 = 15 nM T92521 CS03BA 6255462 IC50 = 800 nM T92521 CTG9I2 6258621 IC50 = 32 nM T92521 CR8P9W 6262995 IC50 = 48 nM T92521 C2U5JS 6296346 IC50 = 2600 nM T92521 CX59ZP 6971167 IC50 = 690 nM T92521 CM3FR9 7020615 Ki = 670 nM T92521 CWX15G 7514880 IC50 = 96 nM T92521 CY8US6 7946380 IC50 = 112 nM T92521 CSR2O3 8854122 IC50 = 120 nM T92521 CJH57U 8854335 IC50 = 4 nM T92521 CKA23N 9817804 IC50 = 17600 nM T92521 CXNV47 9818893 IC50 = 3200 nM T92521 CW9AH0 9972900 IC50 = 130 nM T92521 CQ8P3D 9973392 IC50 = 90 nM T92521 CT0J8W 10017674 IC50 = 620 nM T92521 CEV95P 10059170 IC50 = 30 nM T92521 C4A5SP 10379988 IC50 = 5210 nM T92521 C8E1KG 10380891 IC50 = 130 nM T92521 C6TE5G 10490229 IC50 = 300 nM T92521 C6UX4J 10633725 IC50 = 7000 nM T92521 CA82YQ 10704488 IC50 > 20000 nM T92521 CHL7C6 10752544 IC50 = 493 nM T92521 CBX64S 10846871 IC50 = 30 nM T92521 CW8I1M 11055725 IC50 = 4900 nM T92521 C4S3NP 11066044 IC50 = 390 nM T92521 CH61UW 11128957 IC50 > 20000 nM T92521 C2KE8Z 11130361 IC50 = 370 nM T92521 CSQ18T 11206660 Ki = 12000 nM T92521 CV1SD9 11208566 IC50 = 220 nM T92521 COHR75 11266772 IC50 = 21.6 nM T92521 CBEJ76 11347335 IC50 = 0.49 nM T92521 C4O8WG 11347336 IC50 = 4.2 nM T92521 CJ3LG8 11392135 IC50 = 2.7 nM T92521 C41GFC 11808336 IC50 = 97 nM T92521 C9TC3K 12136078 Ki = 2300 nM T92521 CSIG61 12412902 Ki = 180 nM T92521 CPNR74 12921022 IC50 = 16.7 nM T92521 CJX18P 13267935 Ki = 28000 nM T92521 C0FY4P 13615899 IC50 = 65 nM T92521 CE2JH5 13893963 IC50 = 140 nM T92521 CT19BZ 14026465 IC50 = 76.9 nM T92521 CIF90V 14434140 IC50 = 15 nM T92521 C7BWX3 14914715 IC50 = 222 nM T92521 C5B9KO 15252040 IC50 = 187 nM T92521 CTWY65 15549947 IC50 = 120 nM T92521 C38JKM 15556475 IC50 = 55.4 nM T92521 C1XJU3 15556476 IC50 = 46.6 nM T92521 C8WLJ1 15723463 IC50 = 7.8 nM T92521 CN76ZE 16737013 IC50 = 666 nM T92521 C8D4PX 17408359 IC50 = 64 nM T92521 C2HFY3 19553304 IC50 = 31 nM T92521 CD13BU 19560590 IC50 = 130 nM T92521 CFQ10V 21239772 IC50 = 135 nM T92521 C3BXE1 22983886 IC50 = 3400 nM T92521 CU8C0I 24233261 IC50 = 189 nM T92521 CM51PG 24721239 IC50 = 3.8 nM T92521 CE63OB 40700807 IC50 = 23 nM T92521 CHW3D1 40700815 IC50 = 59 nM T92521 CNO97U 44255810 IC50 = 8500 nM T92521 C3VLK2 44318917 IC50 = 140 nM T92521 C7LVC8 44319156 IC50 = 140 nM T92521 CWCB79 44319159 IC50 = 80 nM T92521 C8JI0A 44319169 IC50 = 2402 nM T92521 CVNM65 44347296 IC50 = 2 nM T92521 C4HOT5 44470750 IC50 = 301 nM T92521 CSW2X1 44591967 IC50 = 137 nM T92521 CPG61Y 44718445 IC50 > 20000 nM T92521 CHB43E 45028066 IC50 = 240 nM T92521 CQK92W 46931209 IC50 = 1.77 nM T92521 CUY75P 49865518 IC50 = 539.8 nM T92521 CKG5Z8 66553582 IC50 = 2000 nM T92521 CR03HY 66553583 IC50 = 1100 nM T92521 CMW4E6 66553584 IC50 = 1000 nM T92521 C7E2SJ 66553585 IC50 = 900 nM T92521 CRMG97 66553586 IC50 = 500 nM T92521 CFP95J 66553587 IC50 = 300 nM T92521 CF9DT8 69248278 IC50 = 300 nM T92521 CJ1FN6 70682593 Ki = 41 nM T92521 C3OZ0N 70682594 IC50 = 1500 nM T92521 C5UC0Z 70688284 IC50 = 336 nM T92521 C3PJX7 70695190 Ki = 30 nM T92521 CQWA13 70695191 IC50 = 5500 nM T92521 C0G3TY 70697234 IC50 = 1100 nM T92521 C5TB7D 71364816 IC50 = 3.5 nM T92521 CI0VR5 71662265 Ki = 53 nM T92521 CZ01TB 71662427 Ki = 5.6 nM T92521 C61BEP 71738859 IC50 = 310 nM T92521 CU4Q1J 73774541 IC50 = 18000 nM T92521 C89FRV 76311181 IC50 = 4 nM T92521 CF07EK 76313382 IC50 > 20000 nM T92521 COX36R 76314785 IC50 = 4170 nM T92521 CJO15N 76316894 IC50 > 20000 nM T92521 C3OP2B 76319044 IC50 = 22 nM T92521 CXVK96 76322062 IC50 = 210 nM T92521 C76UKL 76333454 IC50 > 20000 nM T92521 CT73EY 76336509 IC50 = 4440 nM T92521 C3H5XR 82639722 IC50 = 170 nM T92521 C3Q6VU 85977688 IC50 = 48.4 nM T92521 CQ96AK 90666858 IC50 = 98.2 nM T92521 CL1Y7W 90666859 IC50 = 350 nM T92521 CZU4F0 90666860 IC50 = 192 nM T92521 CQ15SP 90666861 IC50 = 78.4 nM T92521 CI5V3O 90666862 IC50 = 148 nM T92521 CP0DS8 90666863 IC50 = 420 nM T92521 CJA06R 91755082 Ki = 20400 nM T92521 C3I0AL 102004360 IC50 = 19.6 nM T92521 C5QM6D 102351043 IC50 = 90 nM T92521 C87GEW 102435977 IC50 = 900 nM T92521 CLM53V 118491075 IC50 = 133 nM T92521 C9TAD2 118491240 IC50 = 106 nM T92521 C8PU5O 118491249 IC50 = 610 nM T92521 C3KAO6 118491258 EC50 = 10000 nM T92521 CINA28 118492166 IC50 = 48 nM T92521 C2M1TV 118735488 IC50 = 0.2 nM T92521 C7QP3F 118735489 IC50 = 0.2 nM T92521 CA3HP5 118735490 IC50 = 0.043 nM T92521 CZSX60 118735516 IC50 = 0.3 nM T92521 CXO96N 118735517 IC50 = 1.1 nM T92521 CR41NX 118735518 IC50 = 0.3 nM T92521 CVUY89 118735519 IC50 = 0.2 nM T92521 CX4A1O 118735520 IC50 = 9 nM T92521 CT58CZ 118735521 IC50 = 1.1 nM T92521 CU60HF 118735522 IC50 = 2.5 nM T92521 CJ41PI 118735523 IC50 = 9.8 nM T92521 CH70UE 118735524 IC50 = 771.4 nM T92521 C0V2KO 118735525 IC50 > 100000 nM T92521 CA0BG3 118735526 IC50 = 642.9 nM T92521 CY6M3U 118735527 IC50 = 62.9 nM T92521 CIL7X8 118735528 IC50 = 2.3 nM T92521 CA59RL 118735529 IC50 = 1.2 nM T92521 CK1Z3T 118735530 IC50 = 0.3 nM T92521 C8M0UY 118735531 IC50 = 0.8 nM T92521 CJ7M5Y 118735532 IC50 = 1.6 nM T92521 CL6QK3 118735533 IC50 = 3.5 nM T92521 CCH76J 118735534 IC50 = 5 nM T92521 CIX1W5 118735535 IC50 = 98.4 nM T92521 CY4Q8E 118735537 IC50 = 114.5 nM T92521 C4N0LJ 118735539 IC50 = 37.02 nM T92521 C9FSN4 118735541 IC50 = 68.81 nM T92521 CP41AT 118735544 IC50 = 25300 nM T92521 CQ70PY 122184915 Ki = 100 nM T92521 CZ5PR4 122184916 Ki = 120 nM T92521 CK4H2U 122184917 Ki = 480 nM T92521 CFI8N5 122184918 Ki = 5040 nM T92521 C4RCQ2 122184919 Ki = 21200 nM T92521 C51ZRN 122184920 Ki = 4620 nM T92521 C5L3HV 122184965 Ki = 22600 nM T92521 CA07CS 122184966 Ki = 46800 nM T92521 C5YV0E 122184967 Ki = 46600 nM T92521 CZG0V7 122184968 Ki = 30100 nM T92521 CWDI07 127037076 IC50 = 1500 nM T92521 CCJX69 127041842 IC50 > 20000 nM T92521 COH43C 129678161 IC50 = 151.3 nM T92521 CR3X8L 132544693 IC50 = 90.2 nM T92521 CIS9K5 135421564 IC50 = 3 nM T92521 CSVG36 135427256 IC50 = 170 nM T92521 CVB6W9 135492463 IC50 = 37 nM T92521 CVS8F5 136026475 IC50 = 160 nM T92521 C4HJ7D 136044076 IC50 = 54 nM T92521 C95TJH 136632047 IC50 = 141 nM T92521 CI94YQ 136982007 IC50 = 2 nM T92521 CO7YM9 137348938 IC50 = 4.4 nM T92521 C6JO4G 137631841 IC50 > 20000 nM T92521 CW32LA 137634245 IC50 = 162 nM T92521 CIUF50 137634527 IC50 > 5000 nM T92521 CLC5K9 137634802 IC50 = 5.6 nM T92521 CWL25K 137636500 IC50 = 0.52 nM T92521 C2Y9HF 137638913 IC50 > 20000 nM T92521 CO8V4W 137642907 IC50 > 20000 nM T92521 CJT81N 137643054 IC50 > 20000 nM T92521 C1FU3P 137643308 IC50 > 20000 nM T92521 CN97GA 137645181 IC50 = 120 nM T92521 CU47YW 137646415 IC50 > 20000 nM T92521 C5IHS8 137646440 IC50 = 2700 nM T92521 C5AT7D 137649062 IC50 = 9200 nM T92521 CB61UY 137658460 IC50 > 20000 nM T92521 CG96FH 137658637 IC50 = 4 nM T92521 C06DSZ 144648669 IC50 = 4.8 nM T92521 C1UCX0 144953608 IC50 = 3810 nM T92521 C9GRB2 144953612 IC50 = 2920 nM T92521 CV4X5P 144953614 IC50 = 8620 nM T92521 CWN7P3 145952241 IC50 = 32 nM T92521 CZW27Y 145957956 IC50 = 11 nM T92521 CNG9W8 145959850 IC50 = 63 nM T92521 C26ALC 145968480 IC50 = 370 nM T92521 CE5IU1 145972644 IC50 = 120 nM T92521 C2SN5M 145976850 IC50 = 540 nM T92521 CI4ZQ1 155510681 IC50 = 3.2 nM T92521 CCQW36 155511603 IC50 = 90.3 nM T92521 CJSF06 155513229 IC50 = 40.5 nM T92521 C06OGW 155514987 IC50 = 38.8 nM T92521 CP3CG5 155518163 IC50 > 1000 nM T92521 CGZK13 155518556 IC50 = 89.7 nM T92521 CPK3U6 155519244 IC50 = 4 nM T92521 CVB16D 155523847 IC50 = 4.9 nM T92521 C8Z5TR 155525476 IC50 = 4.1 nM T92521 C29OTC 155527077 IC50 = 10.4 nM T92521 CA13JV 155529320 IC50 = 222.9 nM T92521 CD5RZ1 155531248 IC50 = 13.3 nM T92521 CA6DT8 155532021 IC50 = 8 nM T92521 CF8X4L 155533097 IC50 = 51.4 nM T92521 CC7U2N 155534507 IC50 = 63.8 nM T92521 C2GSK9 155534524 IC50 = 24.3 nM T92521 C8B3ZE 155534785 IC50 = 51.9 nM T92521 CO0H8P 155534820 IC50 = 250.4 nM T92521 C6MEB0 155536583 IC50 = 112.4 nM T92521 CT01QV 155537114 IC50 = 2.6 nM T92521 C4HYA1 155537214 IC50 = 1.6 nM T92521 C39JUR 155539220 IC50 = 1.8 nM T92521 CX9HN6 155540486 IC50 = 18.8 nM T92521 CX9T4A 155541298 IC50 = 47.7 nM T92521 CFH72X 155541389 IC50 = 81.9 nM T92521 CO5NZ0 155543459 IC50 = 51.8 nM T92521 C9RPB5 155546584 IC50 = 3.6 nM T92521 CH78RF 155547056 IC50 = 2 nM T92521 C2NI3C 155550109 IC50 = 3.9 nM T92521 CFG8W1 155550859 IC50 = 48.31 nM T92521 CO8LW4 155551203 IC50 = 3.2 nM T92521 CIR3V2 155551390 IC50 = 13.4 nM T92521 C2VLU5 155551528 IC50 > 5000 nM T92521 CFVN26 155552491 IC50 = 103.6 nM T92521 CW72FS 155552958 IC50 = 4.2 nM T92521 CQRJ62 155555492 IC50 = 9.1 nM T92521 CZ8OV2 155555692 IC50 = 9.4 nM T92521 CO3X8Q 155557047 IC50 = 5 nM T92521 CW9YE5 155557609 IC50 = 4.1 nM T92521 CP7R2X 155558740 IC50 > 5000 nM T92521 COSR91 155558908 IC50 = 10.6 nM T92521 CQAI41 155561729 IC50 = 90.2 nM T92521 CAWT92 155562817 IC50 = 23.5 nM T92521 COG7H9 155563270 IC50 = 66.1 nM T92521 C1N8OX 155564817 IC50 > 5000 nM T92521 CJZ92T 155566955 IC50 = 24.6 nM T92521 D00AII 5281727 Ki = 900 nM T92521 D00LMG 5281697 Ki = 220 nM T92521 D00RFY 5281612 Ki = 16 nM T92521 D00RIX 5280443 Ki = 64 nM T92521 D00YEV 5281605 Ki = 260 nM T92521 D01FGM 5280666 IC50 = 19.7 nM T92521 D01FJE 160481 IC50 = 1024 nM T92521 D01KKU 5281894 IC50 = 250 nM T92521 D01UYI 5281607 Ki = 16 nM T92521 D03IQX 11415057 IC50 = 3.3 nM T92521 D04DYO 5281666 IC50 = 6 nM T92521 D06PZE 5281699 IC50 = 20 nM T92521 D06VXW 10105252 IC50 = 2100 nM T92521 D06YKU 68112 IC50 = 210 nM T92521 D06ZRX 5281717 IC50 = 34000 nM T92521 D07YDN 5281654 Ki = 3 nM T92521 D08AIJ 440735 IC50 = 1284 nM T92521 D09ROW 10212 Ki = 1000 nM T92521 D0AS0V 10141 IC50 > 10000 nM T92521 D0B5GC 11349 IC50 = 90 nM T92521 D0CR8V 73635 IC50 = 240 nM T92521 D0F5EI 10017019 IC50 = 213 nM T92521 D0G3TK 5280863 Ki = 43 nM T92521 D0I7GE 11790 IC50 = 4 nM T92521 D0J9OG 2321450 IC50 = 670 nM T92521 D0KG0Z 11471812 IC50 = 2.2 nM T92521 D0M7BR 5280378 Ki = 3700 nM T92521 D0NS1S 5280442 Ki = 7 nM T92521 D0O9NE 5388063 IC50 = 790 nM T92521 D0P0IE 10205 IC50 = 6150 nM T92521 D0Q4GJ 323484 IC50 = 6.2 nM T92521 D0S0RK 10680 IC50 = 600 nM T92521 D0S9YX 5280373 Ki = 1900 nM T92521 D0T3PW 5281672 Ki = 27 nM T92521 D0T9DI 3163532 IC50 = 9.3 nM T92521 D0T9IK 11957947 IC50 = 460 nM T92521 D0U5LL 2543 Ki = 148 nM T92521 D0XJ7I 6683 Ki = 700 nM T92521 D0Y7HG 5281616 IC50 = 25 nM T92521 D0Z1AL 9834747 IC50 = 2 nM T69991 D02KKA 24856436 IC50 = 101 nM T69991 D0H8KG 5311382 IC50 = 165 nM T69991 CU5B1Z 4369491 IC50 = 97 nM T69991 C3P8CG 5327885 IC50 = 2600 nM T69991 C4CWI1 5327918 IC50 = 32 nM T69991 CE15KX 9847909 IC50 = 57.54 nM T69991 CGW03A 9975362 IC50 = 180 nM T69991 CWD27O 9976672 IC50 = 33 nM T69991 CZ2F6K 9976901 IC50 = 12.02 nM T69991 CQ0SW7 9978312 IC50 = 23 nM T69991 CG4M8W 9980097 IC50 = 33 nM T69991 CPM0D4 9981170 IC50 = 57 nM T69991 CG7MA0 9997535 IC50 = 70 nM T69991 CD1O6A 10000495 IC50 = 50 nM T69991 CLRN75 10001302 IC50 = 53 nM T69991 CI63HK 10001419 IC50 = 44.67 nM T69991 C0XNP5 10005624 IC50 = 34.67 nM T69991 C0UK4L 10008287 IC50 = 7 nM T69991 CE63WU 10022438 IC50 = 57 nM T69991 C0GMQ1 10022580 IC50 = 41.69 nM T69991 CZF32P 10022581 IC50 = 22.91 nM T69991 CCP9A1 10043931 IC50 = 24 nM T69991 CAZ8D2 10046459 IC50 = 21 nM T69991 CV2Y8H 10051869 IC50 = 35 nM T69991 C6PXJ7 10065463 IC50 = 141.25 nM T69991 CSY3B7 10071975 IC50 = 7.943 nM T69991 CNZ28P 10098763 IC50 = 14 nM T69991 CCQP92 10248686 IC50 = 25 nM T69991 CNQH37 10253652 IC50 = 21 nM T69991 CO8N7L 10318383 IC50 = 15 nM T69991 C3PV5R 10318616 IC50 = 28 nM T69991 C8C2TF 10319524 IC50 = 48.98 nM T69991 C83YTG 10319891 IC50 = 58.88 nM T69991 CX5K6W 10337485 IC50 = 210 nM T69991 C0A3KS 10342897 IC50 = 9 nM T69991 C7I1GX 10343927 IC50 = 13 nM T69991 C1EYA2 10364585 IC50 = 30 nM T69991 C6G9VY 10369451 IC50 = 19 nM T69991 CHN1P0 10384072 IC50 = 11 nM T69991 C9NOZ2 10385019 IC50 = 44.67 nM T69991 C2G3DY 10386664 IC50 = 23 nM T69991 C0UJ5R 10389002 IC50 = 13 nM T69991 CP5IH6 10390085 IC50 = 15.85 nM T69991 CK4CE8 10405212 IC50 = 67 nM T69991 C84OIA 10406993 IC50 = 46.77 nM T69991 C2VR3A 10410783 IC50 = 23 nM T69991 C29BMY 10413815 IC50 = 59 nM T69991 CEF98R 10413846 IC50 = 9 nM T69991 CH8KM7 10414039 IC50 = 12 nM T69991 C5P1XN 10431859 IC50 = 18 nM T69991 CO7Q6H 10434889 IC50 = 54 nM T69991 COP9B6 10435655 IC50 = 24 nM T69991 CR4B6L 10450912 IC50 = 75 nM T69991 CGC12F 10451785 IC50 = 830 nM T69991 CE5HU9 10453390 IC50 = 28 nM T69991 C4A9NC 10472653 IC50 = 60 nM T69991 CD25UL 10475362 IC50 = 26.92 nM T69991 CC3DV9 10477305 IC50 = 19.95 nM T69991 CM5WA8 10478085 IC50 = 26.92 nM T69991 CC9WA7 11612456 IC50 = 110 nM T69991 CTSG65 11740347 IC50 = 24 nM T69991 CW4EK0 11740418 IC50 = 28.18 nM T69991 CAOB03 11744406 IC50 = 30 nM T69991 CE1N3Y 11744724 IC50 = 7 nM T69991 CST3M7 11749233 IC50 = 410 nM T69991 CU9RM0 11842834 IC50 = 2300 nM T69991 CGSY90 11842835 IC50 > 50000 nM T69991 CZ23AN 11842836 IC50 = 78 nM T69991 CR25PH 11842837 IC50 = 1600 nM T69991 CYHR74 11842838 IC50 = 2300 nM T69991 C14TDN 11842839 IC50 = 29000 nM T69991 C0X4KO 11842840 IC50 = 1100 nM T69991 CVR2K9 11842841 IC50 = 269.15 nM T69991 C1Z3RW 11842842 IC50 = 109.65 nM T69991 CG3NR8 11842843 IC50 = 28.84 nM T69991 C05ALU 11842844 IC50 = 180 nM T69991 CL3Q1S 11842845 IC50 = 13000 nM T69991 CULN90 11842846 IC50 = 575.44 nM T69991 CCG3Q9 11842994 IC50 > 50000 nM T69991 CUMC05 11842995 IC50 = 37000 nM T69991 C87DLM 11842996 IC50 > 50000 nM T69991 CQ6H1Z 11842997 IC50 = 330 nM T69991 CKDH12 11842998 IC50 = 510 nM T69991 C2EXY1 11842999 IC50 = 446.68 nM T69991 C54KPJ 11843000 IC50 = 160 nM T69991 C63JZI 11843001 IC50 = 257.04 nM T69991 CI6DR2 11843002 IC50 = 63 nM T69991 CE71YT 11843003 IC50 = 170 nM T69991 CSW06V 11843143 IC50 = 220 nM T69991 C0QY1S 11843144 IC50 = 229.09 nM T69991 CH29RF 11843145 IC50 = 870 nM T69991 CXB5U7 11843146 IC50 = 40000 nM T69991 CA2JS9 11843147 IC50 = 620 nM T69991 CQF74N 11843148 IC50 = 16000 nM T69991 C1RB0T 11843149 IC50 = 3300 nM T69991 CRQ01W 11843150 IC50 = 1200 nM T69991 CHG2O7 11843287 IC50 = 3600 nM T69991 C6AR4K 11843288 IC50 = 12000 nM T69991 C60DPL 11843289 IC50 = 151.36 nM T69991 C5ZF4Y 11843290 IC50 = 489.78 nM T69991 C94ELW 11843291 IC50 = 19.95 nM T69991 C2YV6D 11843292 IC50 = 954.99 nM T69991 C9K2MI 11843293 IC50 = 19 nM T69991 C2KVO5 11843428 IC50 = 42 nM T69991 CK1BJ7 11843429 IC50 = 38 nM T69991 C36FSN 11843430 IC50 = 812.83 nM T69991 C3O4LX 11843431 IC50 = 10000 nM T69991 CE5O9M 11843432 IC50 = 150 nM T69991 CRZO78 11844343 IC50 = 309.03 nM T69991 C43YKI 11844344 IC50 = 430 nM T69991 C6ET8L 11844345 IC50 = 140 nM T69991 CVNB38 11844346 IC50 = 130 nM T69991 CI3KG0 11844347 IC50 = 9700 nM T69991 C0I2DQ 11844478 IC50 = 4000 nM T69991 C1M3LN 11844479 IC50 = 20000 nM T69991 C1JMO5 11844480 IC50 = 2800 nM T69991 CFS47B 11844481 IC50 > 50000 nM T69991 CR48MI 11844482 IC50 = 3900 nM T69991 CYUK21 11844483 IC50 = 640 nM T69991 CWI7A5 11844484 IC50 = 33 nM T69991 CU72HA 11844608 IC50 = 151.36 nM T69991 C4IM8Z 11844609 IC50 = 575.44 nM T69991 CK7O0V 11844610 IC50 = 190 nM T69991 C3X5WY 11844611 IC50 = 570 nM T69991 C95MUX 11844612 IC50 = 218.78 nM T69991 CE50UF 11844613 IC50 = 55 nM T69991 CY2XW1 11844614 IC50 > 50000 nM T69991 CM0V7X 11844749 IC50 = 4400 nM T69991 C2A4QM 11844750 IC50 = 4365.16 nM T69991 CD45ER 11844751 IC50 = 89 nM T69991 CTW53J 11844752 IC50 = 300 nM T69991 CE1L7P 11844753 IC50 = 730 nM T69991 C51FQS 11844754 IC50 > 50000 nM T69991 C5Q1OC 11844755 IC50 = 1819.7 nM T69991 C5VPH9 16129448 IC50 = 3650 nM T69991 C62KMD 21980334 IC50 = 19 nM T69991 C05BIJ 21980353 IC50 = 35 nM T69991 C5H0QS 21980362 IC50 = 81.28 nM T69991 C13WHU 21980365 IC50 = 58 nM T69991 CV67ME 21980368 IC50 = 40000 nM T69991 CQY89R 21980377 IC50 = 290 nM T69991 C39NXD 21980383 IC50 = 75 nM T69991 CX16UW 21980406 IC50 = 93 nM T69991 C75ZLY 21980427 IC50 = 18 nM T69991 CA6X4C 21980437 IC50 = 280 nM T69991 CSLM60 21980447 IC50 = 24 nM T69991 C0H5VE 21980448 IC50 = 33 nM T69991 C49MKS 21980471 IC50 = 25.7 nM T69991 C8V4OX 21980483 IC50 = 57 nM T69991 C6SBU7 21980490 IC50 = 67 nM T69991 CX9B0Y 21980491 IC50 = 33.88 nM T69991 CKBM87 21980493 IC50 = 36 nM T69991 CTP3I5 21980497 IC50 = 61.66 nM T69991 C3WF0E 21980518 IC50 = 160 nM T69991 CM9DU4 21980529 IC50 = 100 nM T69991 C9C3RQ 21980545 IC50 = 64 nM T69991 C57WSN 21980557 IC50 = 110 nM T69991 C06IXV 21980575 IC50 = 25.7 nM T69991 CD7YS1 21980580 IC50 = 69 nM T69991 CTAO10 21980612 IC50 = 300 nM T69991 CQI80X 21980631 IC50 = 37 nM T69991 CP7BE6 21980647 IC50 = 50 nM T69991 CZVY24 21980658 IC50 = 110 nM T69991 C13NVO 21980695 IC50 = 15 nM T69991 CE93IF 21980705 IC50 = 64 nM T69991 CA24TJ 21980718 IC50 = 48.98 nM T69991 CM37OL 21980722 IC50 = 24 nM T69991 CT3QM7 21980728 IC50 = 230 nM T69991 C42ZAE 21980797 IC50 = 74 nM T69991 C65TXJ 21980800 IC50 = 92 nM T69991 CT3YR9 21980866 IC50 = 71 nM T69991 C7Z4LB 21980883 IC50 = 140 nM T69991 CU84GQ 21980891 IC50 = 140 nM T69991 CT6K9A 21980919 IC50 = 200 nM T69991 CD5XW2 21980923 IC50 = 30 nM T69991 CT13RA 23627206 IC50 = 15 nM T69991 CP5EL9 24884696 IC50 = 8.913 nM T69991 CTFS94 24884697 IC50 = 15 nM T69991 C70ZFW 24884912 IC50 = 6 nM T69991 C0WG1I 24884913 IC50 = 330 nM T69991 CJ1SQ0 24884914 IC50 = 170 nM T69991 C98IDB 24884915 IC50 = 390 nM T69991 CQ3S5Y 24884916 IC50 = 200 nM T69991 CGN52J 24884917 IC50 = 95.5 nM T69991 C0OJM4 24885126 IC50 = 169.82 nM T69991 C68PXG 24885315 IC50 = 120 nM T69991 CWAL41 24885316 IC50 = 360 nM T69991 CJS47Z 44390480 IC50 = 40 nM T69991 CY69XN 44390494 IC50 > 50000 nM T69991 CJ7Y8H 44390497 IC50 = 540 nM T69991 CZY12Q 44390508 IC50 = 550 nM T69991 CSQ6K8 44390517 IC50 = 1200 nM T69991 CV9G7U 44390841 IC50 = 33000 nM T69991 CS41MX 44390847 IC50 = 40 nM T69991 CX8T5B 44390850 IC50 = 1000 nM T69991 CJ8YW9 44390855 IC50 = 95 nM T69991 C26SVZ 44390856 IC50 = 80 nM T69991 CX5W9U 44390861 IC50 > 50000 nM T69991 CH1OD0 44390864 IC50 = 124 nM T69991 C9P6IZ 44390865 IC50 = 120 nM T69991 C5KCA8 44390870 IC50 = 3700 nM T69991 C94IGM 44390873 IC50 = 142 nM T69991 C20XGS 44390874 IC50 = 190 nM T69991 C36AZP 44390876 IC50 = 3600 nM T69991 CI90EM 44390878 IC50 = 250 nM T69991 C53HZB 44390879 IC50 = 260 nM T69991 CFLT82 44390884 IC50 = 990 nM T69991 C7G5TQ 44390885 IC50 = 90 nM T69991 CQW37J 44390890 IC50 > 50000 nM T69991 C16RTZ 44390897 IC50 = 69 nM T69991 CZG92C 44390900 IC50 = 86 nM T69991 C3NTV0 44390902 IC50 = 140 nM T69991 C2YBV4 44390904 IC50 = 150 nM T69991 CC56GH 44390910 IC50 = 1500 nM T69991 CNC80D 44390912 IC50 = 4500 nM T69991 C7YTI1 44390917 IC50 = 8600 nM T69991 CLHX48 44390921 IC50 = 11000 nM T69991 CR3MT8 44390923 IC50 = 27000 nM T69991 C4L9OX 44390924 IC50 > 50000 nM T69991 CKE4V5 44390925 IC50 > 50000 nM T69991 CD50UY 44390926 IC50 = 74 nM T69991 CD8R3Y 44390929 IC50 > 50000 nM T69991 CFA93D 44390937 IC50 = 9700 nM T69991 C2GDX5 44390940 IC50 = 2400 nM T69991 C42QWB 44390941 IC50 = 1900 nM T69991 C4PNF6 44390942 IC50 = 50000 nM T69991 C2X4CS 44390944 IC50 = 410 nM T69991 CZ51FE 44390947 IC50 = 8600 nM T69991 CO4BV8 44390951 IC50 = 3500 nM T69991 CZRV61 44390953 IC50 = 990 nM T69991 CC29YI 44390956 IC50 > 50000 nM T69991 CF83MW 44390957 IC50 = 220 nM T69991 C2ZT8B 44390958 IC50 > 50000 nM T69991 CV3B4S 44390966 IC50 = 3400 nM T69991 CL2G8H 44390967 IC50 = 31000 nM T69991 CKT7Q6 44390968 IC50 = 41000 nM T69991 C46HTU 44390969 IC50 = 2600 nM T69991 CZT7M1 44390972 IC50 = 580 nM T69991 CPFC56 44390982 IC50 > 50000 nM T69991 CL0H4M 44390985 IC50 = 3200 nM T69991 C6H9GQ 44415009 IC50 = 1100 nM T69991 CRJ8F6 44454116 IC50 = 20 nM T69991 CWZ0L4 44454457 IC50 = 46 nM T69991 C3VRO9 44557921 IC50 > 10000 nM T69991 CE3KW5 44593024 IC50 = 20.89 nM T69991 CWV1M5 44593041 IC50 = 199.53 nM T69991 CQ48WT 44593052 IC50 = 64 nM T69991 CU68TO 44593053 IC50 = 109.65 nM T69991 C4S2JM 44593054 IC50 = 230 nM T69991 CZ8F0K 44593055 IC50 = 141.25 nM T69991 C63DNI 44593056 IC50 = 360 nM T69991 C72WYI 44593057 IC50 = 109.65 nM T69991 CC2YH1 44593070 IC50 = 92 nM T69991 CG46FK 44593071 IC50 = 120 nM T69991 C6V0GO 44593072 IC50 = 280 nM T69991 CX5IF9 44593073 IC50 = 54 nM T69991 CPHN90 44593074 IC50 = 19.05 nM T69991 CTL48U 44593091 IC50 = 288.4 nM T69991 CN3OF9 44593092 IC50 = 36.31 nM T69991 CLE94S 44593110 IC50 = 71 nM T69991 CT1DR8 44593111 IC50 = 64 nM T69991 C50NGF 44593112 IC50 = 59 nM T69991 CFS3A0 44593113 IC50 = 302 nM T69991 CKH0X6 44593114 IC50 = 160 nM T69991 CM1OQ8 44593127 IC50 = 93 nM T69991 CU86TX 44593128 IC50 = 170 nM T69991 C8FT3S 44593145 IC50 = 22.91 nM T69991 CF8MN0 44593194 IC50 = 23.99 nM T69991 C6C4PL 44593195 IC50 = 23.99 nM T69991 CFS47D 44593196 IC50 = 8.913 nM T69991 CI95XQ 44593217 IC50 = 50 nM T69991 CE2S9G 44593218 IC50 = 36.31 nM T69991 C6NV3P 44593239 IC50 = 23.99 nM T69991 C9WUE4 44593260 IC50 = 75 nM T69991 C8UZF1 44593261 IC50 = 18 nM T69991 CHXP96 44593281 IC50 = 23.99 nM T69991 CSTR98 44593282 IC50 = 19.95 nM T69991 CQ8ED9 44593304 IC50 = 140 nM T69991 CU4K3V 44593305 IC50 = 25 nM T69991 C58IVW 44593306 IC50 = 33 nM T69991 CJB6M4 44593307 IC50 = 46 nM T69991 CV53JR 44593308 IC50 = 15 nM T69991 CPFB46 44593325 IC50 = 199.53 nM T69991 CD2K4R 50908681 Ki > 1000000 nM T69991 CM42BY 51000510 Ki > 1000000 nM T69991 C8YE5A 60153266 Ki = 2.3 nM T69991 CU65AC 60168496 Ki = 21 nM T69991 CFZI84 60168590 Ki = 26 nM T69991 CPYH50 60168684 Ki = 8.6 nM T69991 CUIJ08 60169069 Ki = 7.4 nM T69991 C6GN2M 60169070 Ki = 2 nM T69991 CO0QP6 60169337 Ki < 1 nM T69991 C37NKO 67129970 IC50 > 10000 nM T69991 CK80LJ 67130050 IC50 > 10000 nM T69991 CV63UL 67240318 IC50 > 10000 nM T69991 C4WHB2 68193664 Ki = 5.4 nM T69991 C2OL8V 68194699 Ki = 1.2 nM T69991 CF8G3U 68194810 Ki < 1 nM T69991 CZSD28 68194869 Ki < 1 nM T69991 CMW6B3 68194909 Ki < 1 nM T69991 C32IUK 68195012 Ki = 6.2 nM T69991 C8UXP1 68195019 Ki = 87 nM T69991 CLO41Y 68195071 Ki = 6.6 nM T69991 C8RHU9 68195086 Ki = 8.3 nM T69991 CBVH05 68195167 Ki = 5.5 nM T69991 CSO8C6 68195176 Ki = 1.6 nM T69991 CEM54B 68195199 Ki < 1 nM T69991 C2B9PS 68195324 Ki < 1 nM T69991 C7GRV2 68755406 IC50 > 10000 nM T69991 C0HA8V 68783839 IC50 = 2800 nM T69991 CS3PD4 71543379 Ki = 0.2 nM T69991 CQ0AC1 71555192 Ki = 0.3 nM T69991 CQUA08 71555194 Ki = 1 nM T69991 CQGC04 71555272 Ki = 24.4 nM T69991 C9XT6O 71555274 Ki = 0.2 nM T69991 CJ3D7E 71555419 Ki = 1.3 nM T69991 CYI9J4 71724470 Ki = 0.3 nM T69991 C09FKM 71724574 Ki = 0.3 nM T69991 C0JK9Y 71724880 Ki = 0.5 nM T69991 C7S8NW 89511429 Ki = 0.6 nM T69991 C5MY0Z 89511484 Ki = 0.2 nM T69991 CBO8H9 89511537 Ki = 0.3 nM T69991 C2FRY7 89511604 Ki = 0.2 nM T69991 CZ7KB4 89764767 Ki = 0.6 nM T69991 C1TS3Q 118720915 Ki > 3140 nM T69991 C7UMK2 118720916 Ki > 3140 nM T69991 CZ7EX0 136183413 IC50 = 5720 nM T69991 CI1E8V 137634241 IC50 = 9880 nM T69991 CS61AX 137659496 IC50 > 100000 nM T69991 C2MD1Q 155513187 IC50 > 10000 nM T69991 C86HPW 155518524 IC50 = 79000 nM T69991 D0Y3PH 11844342 IC50 = 97 nM T23995 D02UFQ 11620908 IC50 > 10000 nM T23995 D03LWG 53235510 IC50 > 10000 nM T23995 D07EHV 44814409 IC50 = 4100 nM T23995 D09DHT 27924 EC50 = 3190 nM T23995 D0E3TC 44259 IC50 = 1.44 nM T23995 D0MS3Z 16725726 IC50 = 2 nM T23995 D03BNU 59604787 IC50 > 10000 nM T23995 D0T3ME 156422 IC50 > 30000 nM T23995 C8PU1O 188534 Ki = 1.4 nM T23995 C5UM8B 513197 IC50 = 31600 nM T23995 CQ59SY 639665 IC50 > 100000 nM T23995 CMKE97 3071991 IC50 = 453000 nM T23995 C2RA4O 5352033 Ki = 0.11 nM T23995 C0IK9O 9543716 EC50 = 8670 nM T23995 CQD2W7 9935079 IC50 = 65 nM T23995 CP5NJ3 9952970 Ki = 13.2 nM T23995 C0V7UW 9958506 IC50 > 11000 nM T23995 C12COP 9977326 IC50 = 3700 nM T23995 CFK4B1 10000619 IC50 = 110 nM T23995 CZ08EJ 10001382 IC50 = 35 nM T23995 C98KZE 10002960 IC50 = 54 nM T23995 CU3NK5 10045795 IC50 = 210 nM T23995 C48GBP 10046543 IC50 = 210 nM T23995 C7YD1X 10048045 IC50 > 25000 nM T23995 C4EOY0 10048329 IC50 = 1500 nM T23995 C7F0GK 10069466 IC50 = 180 nM T23995 CQ8GZ3 10092284 IC50 = 2500 nM T23995 CJ2M5B 10092312 IC50 = 200 nM T23995 C2O7ZH 10137972 IC50 = 2.1 nM T23995 CZJI60 10141037 IC50 > 10000 nM T23995 C94WRY 10143231 IC50 > 10000 nM T23995 C5P8JC 10206423 IC50 = 835 nM T23995 C2U5AI 10252616 IC50 = 27 nM T23995 C7UC9A 10253430 IC50 = 18 nM T23995 C7SFI1 10296883 IC50 = 1 nM T23995 CI1GH3 10318082 IC50 = 48 nM T23995 CTMH50 10318687 IC50 = 910 nM T23995 C96RXP 10319074 IC50 = 170 nM T23995 CFU38G 10363814 Ki = 358 nM T23995 C3LM2U 10386385 IC50 = 54 nM T23995 C2N5PR 10386615 IC50 = 22 nM T23995 C3RBY8 10395226 Ki = 6.6 nM T23995 C8I7EP 10407691 IC50 = 34 nM T23995 CVZ12K 10407692 IC50 = 39 nM T23995 C6NU1M 10408604 IC50 = 160 nM T23995 CJA79B 10408796 IC50 = 77 nM T23995 CRIQ70 10410919 IC50 = 7 nM T23995 CNL7O0 10410920 IC50 = 8 nM T23995 CQXJ51 10425978 Ki = 61.6 nM T23995 CY9Q5T 10430990 IC50 = 13 nM T23995 CO23BZ 10431115 IC50 = 17 nM T23995 C2SWM0 10431370 IC50 = 85 nM T23995 CIOH31 10431441 IC50 = 42 nM T23995 CGI8B4 10433832 IC50 = 5 nM T23995 C36QRS 10453829 Ki = 167 nM T23995 CZPM04 10456238 IC50 = 39 nM T23995 C1VI3E 10477747 IC50 = 255 nM T23995 C2G5CU 10894726 Ki = 1097 nM T23995 CR47CD 11025838 Ki = 62 nM T23995 C67CSJ 11201611 IC50 = 185 nM T23995 C3ROM0 11247414 IC50 = 216 nM T23995 CRZ38O 11315034 IC50 = 276 nM T23995 C4ON7Z 11362429 IC50 = 12 nM T23995 C3KAC4 11538477 IC50 > 316 nM T23995 C1CD2N 11547825 IC50 = 314 nM T23995 C9OV5S 11561609 IC50 = 101 nM T23995 CD7PF5 11574473 IC50 > 316 nM T23995 CA9XJ2 11604381 IC50 = 21 nM T23995 CI9HQ2 11624816 IC50 > 316 nM T23995 CQ5S3G 11639520 IC50 > 316 nM T23995 CU0E8O 11690457 Ki = 290 nM T23995 CR20HY 11741829 IC50 = 130 nM T23995 CX97TV 11741992 IC50 = 3 nM T23995 CVOQ03 11742057 IC50 = 100 nM T23995 C1GO3E 11743836 IC50 = 12 nM T23995 CP7AH3 11755812 IC50 = 50000 nM T23995 CS36BH 11843159 IC50 > 5000 nM T23995 CTN96I 11851810 IC50 = 0.5 nM T23995 CW53JC 11998038 Ki = 3 nM T23995 CQ39BY 12115602 IC50 = 3.3 nM T23995 C7LB4I 15949613 IC50 > 10000 nM T23995 C86KBM 16123360 IC50 = 75 nM T23995 C68NYP 16123362 IC50 = 100 nM T23995 CMB17Y 16123474 IC50 > 5000 nM T23995 CNF5W8 16123475 IC50 > 5000 nM T23995 CGAB24 16123478 IC50 > 5000 nM T23995 C2O3GT 16123588 IC50 = 1300 nM T23995 C8GTX1 16123589 IC50 = 830 nM T23995 C9P6EB 16123591 IC50 > 5000 nM T23995 CP5T1W 16123594 IC50 = 1800 nM T23995 CV4CF9 16123704 IC50 = 52 nM T23995 C7Q5WR 16123707 IC50 = 570 nM T23995 C8WNA0 16123709 IC50 = 450 nM T23995 CR92JO 16124248 IC50 = 93 nM T23995 CP2M4O 16124345 IC50 = 14 nM T23995 C5VPH9 16129448 IC50 = 7510 nM T23995 CG04RZ 16727123 IC50 = 18 nM T23995 CWH37T 17758574 IC50 > 50000 nM T23995 C59JGV 21080665 IC50 = 640 nM T23995 CG4JD1 21081008 IC50 = 500 nM T23995 C9AVK0 21113469 IC50 = 165 nM T23995 CS15LY 21672114 Ki = 0.16 nM T23995 CZ0X8J 22592015 IC50 > 315 nM T23995 CW6OB1 23627212 IC50 = 0.28 nM T23995 CK73JS 24742033 Ki = 12 nM T23995 C7YG1N 24759534 IC50 = 6600 nM T23995 C2UOE0 24766030 IC50 = 3.8 nM T23995 CJUK39 24770517 Ki = 79 nM T23995 CM28WD 24825721 IC50 = 7.4 nM T23995 CBSX32 24858083 IC50 = 900 nM T23995 CX0O7A 24858085 IC50 > 30000 nM T23995 CHK54R 24858240 IC50 = 80 nM T23995 CPX4U2 24858411 IC50 = 4600 nM T23995 CK20QZ 24859980 IC50 = 3900 nM T23995 CM80XP 24859981 IC50 = 1400 nM T23995 C9SKN0 24859982 IC50 = 1600 nM T23995 CFUY94 24860129 IC50 = 2200 nM T23995 CUL6Z1 24860132 IC50 = 2800 nM T23995 CV1L9B 24860133 IC50 = 160 nM T23995 C1L7UO 24860134 IC50 = 400 nM T23995 C58XGF 24860268 IC50 = 8400 nM T23995 C9F7YH 24860269 IC50 = 470 nM T23995 C9C3VL 24860271 IC50 = 2400 nM T23995 C3LQ2T 24860273 IC50 > 30000 nM T23995 CR0PH4 24865071 IC50 = 63 nM T23995 C9NT5W 24865072 IC50 = 320 nM T23995 C8HG3V 24865073 IC50 = 6300 nM T23995 C2TL9X 24865433 IC50 = 32 nM T23995 CSW5V3 24865437 IC50 = 18 nM T23995 CPGW60 24865438 IC50 = 29 nM T23995 CJ7NM3 24865614 IC50 = 17 nM T23995 CAT18G 24865615 IC50 = 60 nM T23995 CTZP64 24865617 IC50 = 9500 nM T23995 CFE7K0 24865618 IC50 = 190 nM T23995 CO2G8E 24865619 IC50 = 200 nM T23995 C93XKC 24866508 IC50 = 2200 nM T23995 CEP58J 24866676 IC50 = 2000 nM T23995 CPV6Y5 24866677 IC50 = 13 nM T23995 C36PKE 24992835 Ki = 164 nM T23995 C8D7ER 24993153 Ki = 1390 nM T23995 CMP8Z9 24993483 Ki = 3 nM T23995 C3A5BK 24993785 Ki = 4 nM T23995 C3H4TS 24993787 Ki = 182 nM T23995 C2JO7A 24994105 Ki = 67 nM T23995 CVZ5K7 24994106 Ki = 85 nM T23995 CH4RO0 24994728 Ki = 290 nM T23995 C6E9WR 24995040 Ki = 28 nM T23995 CS3Q8B 24995659 Ki = 3 nM T23995 C2WXE1 24995663 Ki = 2 nM T23995 C1ONA4 24996161 IC50 = 141 nM T23995 C6P1CX 25066843 IC50 = 7.5 nM T23995 CDO3X2 25113021 IC50 = 997 nM T23995 CBI73N 25113026 IC50 = 355 nM T23995 C1R0JL 25113028 IC50 = 97 nM T23995 C4KL8Q 25113038 IC50 = 140 nM T23995 CV58WZ 25113039 IC50 > 1000 nM T23995 C8KI1Z 25113050 IC50 > 1000 nM T23995 CTV54O 25123227 IC50 > 10000 nM T23995 CR0S2O 25195244 IC50 = 8.7 nM T23995 CTX60V 25195245 IC50 = 9.2 nM T23995 C6FGQ1 25206346 IC50 > 10000 nM T23995 CRO09K 25211064 IC50 = 27400 nM T23995 C92QDU 42611189 Ki = 14 nM T23995 CU9E4P 42629114 IC50 = 3500 nM T23995 CBP7K1 42633428 Ki = 9 nM T23995 CFT83M 42633778 Ki = 0.3 nM T23995 CW24IK 42633780 Ki = 3 nM T23995 C75GFD 42633960 Ki = 9 nM T23995 CAO2T4 42634832 Ki = 28 nM T23995 C70RVN 42635564 Ki = 3 nM T23995 C13SQT 42635568 Ki = 17 nM T23995 CU3D9V 42635569 Ki = 22 nM T23995 C4UMB7 44158300 Ki = 4 nM T23995 C4G5DI 44158301 Ki = 170 nM T23995 CLW80F 44160269 IC50 = 1.8 nM T23995 C8KNA3 44219632 Ki > 4000 nM T23995 C0VIX4 44219633 Ki = 1800 nM T23995 CEL61X 44229839 IC50 > 10000 nM T23995 CIX8V2 44251637 IC50 = 10 nM T23995 CGH06R 44251772 IC50 = 22 nM T23995 CP89VQ 44251773 IC50 = 11 nM T23995 C4FB3W 44251775 IC50 = 38 nM T23995 CZJO40 44251776 IC50 = 12 nM T23995 CB26IP 44251778 IC50 = 6.4 nM T23995 CM5LK7 44251903 IC50 = 22 nM T23995 CU93BX 44251904 IC50 = 23 nM T23995 CKZ3V2 44251905 IC50 = 3.5 nM T23995 CWUZ68 44251906 IC50 = 8.9 nM T23995 CX4AO2 44251907 IC50 = 3.6 nM T23995 CHW1Y9 44251908 IC50 = 9.3 nM T23995 CX23BG 44252049 IC50 = 6.8 nM T23995 C09WSD 44252050 IC50 = 5.7 nM T23995 C3VQ0G 44252052 IC50 = 19 nM T23995 C9JP5W 44252053 IC50 = 4.9 nM T23995 C7RFS9 44252054 IC50 = 6 nM T23995 C5GV6Y 44252348 IC50 = 71 nM T23995 C1S4EF 44252350 IC50 = 3.6 nM T23995 CNBS25 44252635 IC50 = 90 nM T23995 CCV6J0 44252790 IC50 = 1.2 nM T23995 C9AP1D 44252942 IC50 = 1.5 nM T23995 C9QLC5 44253093 IC50 = 4.9 nM T23995 CWJ81C 44253525 IC50 = 8.3 nM T23995 CT6H2N 44253528 IC50 = 31 nM T23995 CLG7I2 44253664 IC50 = 51 nM T23995 C4JX5O 44253666 IC50 = 2.2 nM T23995 C4DIQ1 44253668 IC50 = 68 nM T23995 C9XVU8 44253795 IC50 = 16 nM T23995 CW4C0S 44253797 IC50 = 3.6 nM T23995 C5QFX6 44263382 IC50 = 52 nM T23995 C8RQU2 44263383 IC50 = 76 nM T23995 CZG81D 44263384 IC50 = 4.8 nM T23995 C6YRP1 44263385 IC50 = 1382 nM T23995 CQ13XB 44291629 Ki = 147.5 nM T23995 CERT91 44291669 Ki = 24.1 nM T23995 CO28BT 44376126 Ki = 0.73 nM T23995 CF02IG 44440481 IC50 = 680 nM T23995 CQ08GM 44440482 IC50 = 4200 nM T23995 C07CGQ 44440483 IC50 = 60 nM T23995 C0M4ZA 44440487 IC50 = 83 nM T23995 CVR8I6 44440490 IC50 = 12000 nM T23995 CDML52 44440491 IC50 = 15 nM T23995 C9M4SQ 44440492 IC50 = 6 nM T23995 CP2G6L 44440493 IC50 = 5 nM T23995 C2PZ3I 44440495 IC50 = 11 nM T23995 CM6U2Z 44440496 IC50 = 46 nM T23995 CTN81L 44440499 IC50 = 400 nM T23995 C8V9RN 44440503 IC50 = 2200 nM T23995 C4VUL9 44440505 IC50 = 5700 nM T23995 C36IRE 44440507 IC50 = 4400 nM T23995 CN87ZC 44440508 IC50 = 460 nM T23995 C6DKM7 44440518 IC50 = 31 nM T23995 C8Z6SD 44440519 IC50 = 94 nM T23995 C6SA9O 44440520 IC50 = 270 nM T23995 CP71LK 44440522 IC50 = 90 nM T23995 CXTL17 44440523 IC50 > 10000 nM T23995 C6ZM5Q 44440524 IC50 > 10000 nM T23995 CXSQ75 44440525 IC50 = 90 nM T23995 CE3HF2 44440526 IC50 > 10000 nM T23995 C52OWK 44440527 IC50 = 450 nM T23995 CM1QS0 44449289 IC50 = 730 nM T23995 CX6P0S 44449321 IC50 = 130 nM T23995 CUW91O 44449323 IC50 = 200 nM T23995 CK0NY3 44449384 IC50 = 3700 nM T23995 CYJ7A5 44449412 IC50 > 5000 nM T23995 CSA78Q 44449413 IC50 > 5000 nM T23995 C3RHP2 44449448 IC50 = 230 nM T23995 CHZ8Y2 44449452 IC50 = 52 nM T23995 CY87UN 44456923 Ki = 51.1 nM T23995 CW0T1S 44456924 Ki = 149 nM T23995 CS2CV1 44456938 Ki = 18.6 nM T23995 CCV59D 44473005 IC50 = 190 nM T23995 CX4V8F 44473006 IC50 = 35 nM T23995 CPZ9N7 44473007 IC50 = 19 nM T23995 CSA97D 44473008 IC50 = 34 nM T23995 C5WL1F 44473009 IC50 = 4 nM T23995 C6K7EH 44473010 IC50 = 2.8 nM T23995 CEG1S5 44473011 IC50 = 0.88 nM T23995 CQ02SK 44473012 IC50 = 5.2 nM T23995 C3MR8S 44473013 IC50 = 140 nM T23995 CXW6I3 44473014 IC50 = 11 nM T23995 C0Y5DZ 44473015 IC50 = 1.3 nM T23995 C46OMR 44473016 IC50 = 16 nM T23995 C5L0HD 44473017 IC50 = 31 nM T23995 CQG9E3 44473018 IC50 = 42 nM T23995 C97KBL 44473019 IC50 = 39 nM T23995 CP38JR 44473020 IC50 = 24 nM T23995 C8ZH6C 44473021 IC50 = 7.4 nM T23995 CLB89J 44473022 IC50 = 120 nM T23995 CA03QZ 44473024 IC50 = 12 nM T23995 C73TDV 44473025 IC50 = 50 nM T23995 C02ZEH 44473028 IC50 = 17 nM T23995 C5QX6O 44511325 IC50 = 4.5 nM T23995 C3VRO9 44557921 IC50 > 10000 nM T23995 C8X1JW 44570801 IC50 = 16 nM T23995 CD9BY2 44570802 IC50 = 84 nM T23995 C5BNG9 44570803 IC50 = 23 nM T23995 CC58RY 44570848 IC50 = 100 nM T23995 CGWK29 44570849 IC50 = 12 nM T23995 CJY8S0 44570884 IC50 = 16 nM T23995 CYS8G0 44573871 IC50 = 270 nM T23995 CVGA49 44573872 IC50 = 1700 nM T23995 C15MRZ 44573873 IC50 = 1700 nM T23995 CTW62U 44573874 IC50 = 14 nM T23995 CEV7S0 44573875 IC50 = 11 nM T23995 CXK5I8 44573898 IC50 = 6.3 nM T23995 C3T1UP 44573899 IC50 = 55 nM T23995 C9RCF2 44573900 IC50 = 120 nM T23995 CM9ZP7 44573901 IC50 = 10.5 nM T23995 COJ5C6 44573902 IC50 = 5.9 nM T23995 C7OGY2 44573903 IC50 = 19 nM T23995 CD65VM 44573904 IC50 = 14 nM T23995 CO18GC 44573905 IC50 = 73 nM T23995 CT58FZ 44574268 IC50 = 740 nM T23995 C96NGB 44574269 IC50 = 10.6 nM T23995 C10YAL 44574270 IC50 = 5.3 nM T23995 C7C0FA 44574271 IC50 = 260 nM T23995 C3LKQ1 44574272 IC50 = 27 nM T23995 C26CFS 44574273 IC50 = 5.6 nM T23995 CPG36C 44574310 IC50 = 36 nM T23995 C8OF9M 44574311 IC50 = 82 nM T23995 CAJY35 44574312 IC50 = 20 nM T23995 CF02XQ 44574313 IC50 = 33 nM T23995 C60ZRC 44578247 IC50 = 58 nM T23995 C6B1NX 44578248 IC50 = 22 nM T23995 C3YDK6 44578249 IC50 = 3.5 nM T23995 CD2B4I 44578250 IC50 = 130 nM T23995 C7GDT1 44578680 IC50 = 41 nM T23995 C5AC1P 44578718 IC50 = 180 nM T23995 CL6I2W 44578719 IC50 = 170 nM T23995 C0E3VD 44578720 IC50 = 48 nM T23995 CSYM46 44578721 IC50 = 53 nM T23995 C8TUL6 44578755 IC50 = 88 nM T23995 CT0WO1 44578756 IC50 = 43 nM T23995 CK23LX 44578757 IC50 = 12 nM T23995 C8AD1R 44578758 IC50 = 1.6 nM T23995 C01KPH 44578813 IC50 = 2 nM T23995 C67MLJ 44578814 IC50 = 15 nM T23995 CCY0X5 44578815 IC50 = 110 nM T23995 C0KM7V 44578816 IC50 = 48 nM T23995 CMG72K 44578839 IC50 = 150 nM T23995 C34SOM 44578840 IC50 = 100 nM T23995 C98BRO 44578841 IC50 = 370 nM T23995 CRNT03 44578842 IC50 = 250 nM T23995 C5Z3LI 44591740 IC50 > 30000 nM T23995 CI7MN3 44621943 Ki = 50 nM T23995 C1V6TC 44622679 Ki = 60 nM T23995 CPTY61 44626360 IC50 = 5.3 nM T23995 C06WDZ 45107770 Ki = 2 nM T23995 C7BQ2T 45108044 Ki = 5 nM T23995 C46FDT 45108081 Ki = 15 nM T23995 C16IEQ 45108117 Ki = 12 nM T23995 C8GFI2 45108120 Ki = 68 nM T23995 CC95PQ 45375865 IC50 = 0.49 nM T23995 CEOQ27 45375866 IC50 = 0.44 nM T23995 C6E2SC 45482700 IC50 > 10000 nM T23995 CZXH74 45482750 IC50 > 10000 nM T23995 C9VJH6 45484979 IC50 = 65 nM T23995 C0Y1ZH 45484983 IC50 = 3.6 nM T23995 CM6ZH3 45484989 IC50 = 77 nM T23995 C1T3JI 45484990 IC50 = 13 nM T23995 C4P3XB 45484994 IC50 = 4.7 nM T23995 CR52GN 45485014 IC50 = 440 nM T23995 CXA0O7 45485015 IC50 = 34 nM T23995 C84AUV 45485016 IC50 = 9.1 nM T23995 CG97AV 45485017 IC50 = 79 nM T23995 C8BQ5R 45485037 IC50 = 26 nM T23995 C8M5XT 45485046 IC50 = 4700 nM T23995 C3NYJ6 45485051 IC50 = 360 nM T23995 CA5VN0 45485052 IC50 = 8.2 nM T23995 C3RDZ0 45485058 IC50 = 70 nM T23995 CM93TU 45485059 IC50 = 7 nM T23995 CTK16A 45485067 IC50 = 34 nM T23995 CNPW65 45485068 IC50 = 13 nM T23995 CEY2C0 45485076 IC50 = 7.6 nM T23995 C2S1PV 45485082 IC50 = 190 nM T23995 C5S8MA 45485083 IC50 = 4.7 nM T23995 CSA2U3 45485596 IC50 = 1.7 nM T23995 CF8U6I 45485719 IC50 = 1.4 nM T23995 CX7I1G 45485730 IC50 = 23 nM T23995 CP1TD8 45485731 IC50 = 1.3 nM T23995 CSC38R 45485732 IC50 = 6.4 nM T23995 C3ZHD5 45485733 IC50 = 1.6 nM T23995 CJ94MU 45485734 IC50 = 2.3 nM T23995 C3QJ2U 45485738 IC50 = 2.9 nM T23995 C6LT4C 45485739 IC50 = 13 nM T23995 C2P3WG 45485740 IC50 = 1.5 nM T23995 CS1R6E 45485748 IC50 = 0.48 nM T23995 CZYD36 45485761 IC50 = 2.5 nM T23995 C2B5JI 45485762 IC50 = 2.4 nM T23995 CUJ6X4 45485765 IC50 = 15 nM T23995 CS1K2D 45485766 IC50 = 13 nM T23995 C03NFZ 45485774 IC50 = 6.1 nM T23995 C6O5BP 45485797 IC50 = 0.67 nM T23995 CD3GS6 45487537 IC50 = 12 nM T23995 C0ATH1 45487554 IC50 = 7.8 nM T23995 CTR3P4 45487555 IC50 = 7.5 nM T23995 CHT58B 45487559 IC50 = 38 nM T23995 CTDV41 45487560 IC50 = 190 nM T23995 CFV38T 45487561 IC50 = 41 nM T23995 CW3F7U 45487562 IC50 = 35 nM T23995 C5X8YN 45487570 IC50 = 8.4 nM T23995 CU2J5S 45487571 IC50 = 6.9 nM T23995 CA0CB9 45487572 IC50 = 42 nM T23995 CO0X4N 45487573 IC50 = 1.3 nM T23995 C6AHT9 45487574 IC50 = 2.4 nM T23995 CE3F2I 45487575 IC50 = 3.5 nM T23995 CI24NY 45487588 IC50 = 200 nM T23995 CRJ5X1 45487595 IC50 = 5 nM T23995 CL3K8H 45487596 IC50 = 3 nM T23995 C8HN1Y 45487597 IC50 = 6.1 nM T23995 CCV15K 45487611 IC50 = 9 nM T23995 C76RIH 45487622 IC50 = 23 nM T23995 C5CLP8 45487627 IC50 = 4.9 nM T23995 CW42YX 45487634 IC50 = 4.5 nM T23995 CUA97D 46209401 IC50 > 10000 nM T23995 C6SL3O 46227444 IC50 = 51 nM T23995 CB3I2J 46227490 IC50 = 46 nM T23995 C8UJT1 46227519 IC50 = 57 nM T23995 CQW97N 46846072 IC50 = 1.1 nM T23995 C7H4YM 46865419 IC50 > 10000 nM T23995 CKR46X 46879514 IC50 = 23 nM T23995 CCS06U 46879515 IC50 = 6 nM T23995 CQ1XO5 46879516 IC50 = 12 nM T23995 CB6DH0 46879555 IC50 = 5.4 nM T23995 CF04OQ 46879556 IC50 = 11 nM T23995 CP3K1R 46879557 IC50 = 8.7 nM T23995 CN90TO 46879558 IC50 = 350 nM T23995 C7H9NW 46879602 IC50 = 410 nM T23995 CYW53O 46879603 IC50 = 121 nM T23995 CWJH34 46879604 IC50 = 6 nM T23995 CNUT90 46879605 IC50 = 3 nM T23995 CR14YD 46879645 IC50 = 2.4 nM T23995 C8DH4B 46879687 IC50 = 4.8 nM T23995 CU51HD 46879688 IC50 = 9.3 nM T23995 CJV29C 46879689 IC50 = 21 nM T23995 CZXU95 46879733 IC50 = 68 nM T23995 CS0NZ6 46879734 IC50 = 7.9 nM T23995 CRV8H5 46879735 IC50 = 6.2 nM T23995 C0AW5F 46879777 IC50 = 4.3 nM T23995 CL6GX0 46879778 IC50 = 4.4 nM T23995 CF8OR3 46881461 IC50 = 0.32 nM T23995 CLC24S 46881462 IC50 = 1.4 nM T23995 CN04PB 46881504 IC50 = 9.9 nM T23995 COZS08 46881505 IC50 = 1.9 nM T23995 CARX78 46881506 IC50 = 14 nM T23995 CC9F7R 46881553 IC50 = 4 nM T23995 C8DS7P 46881554 IC50 = 4.1 nM T23995 CWP05I 46881555 IC50 = 1.3 nM T23995 C2LF8C 46881556 IC50 = 5.5 nM T23995 CRVO58 46881593 IC50 = 4.7 nM T23995 CF5M1N 46881594 IC50 = 5.2 nM T23995 CRC2J7 46881595 IC50 = 4.9 nM T23995 C4XBI1 46881640 IC50 = 2.9 nM T23995 CP4F9B 46881641 IC50 = 1.5 nM T23995 C5W8KJ 46881678 IC50 = 56 nM T23995 C8DBP9 46881679 IC50 = 14 nM T23995 C0TE7Y 46881680 IC50 = 2.8 nM T23995 C0NI6L 46881681 IC50 = 31 nM T23995 CVG0L2 46881723 IC50 = 6.2 nM T23995 CKG50T 46881724 IC50 = 3.2 nM T23995 CQN09T 46881725 IC50 = 1.5 nM T23995 CW37OB 46881726 IC50 = 4.3 nM T23995 C9YGL1 46881774 IC50 = 0.84 nM T23995 CH4UA0 46881775 IC50 = 2.1 nM T23995 CEAZ53 46881776 IC50 = 0.65 nM T23995 C1IGH5 46881777 IC50 = 4.2 nM T23995 CSV5B9 46901859 IC50 = 77 nM T23995 C7YJ2X 46901862 IC50 = 109 nM T23995 C1NKE3 46905987 IC50 = 98 nM T23995 CQE9D1 50925411 IC50 = 68 nM T23995 CEQN27 52936621 Ki > 2000 nM T23995 CHP06V 52948258 Ki = 8.1 nM T23995 CR93CL 53308750 Ki = 0.1 nM T23995 C0SWH5 53348216 IC50 > 40000 nM T23995 CD4H3S 53354074 Ki = 0.08 nM T23995 CB32QT 53354075 Ki = 1 nM T23995 C8AB5U 53354478 Ki = 0.1 nM T23995 C8NA4L 53384644 IC50 > 30000 nM T23995 CUY9G2 53473663 IC50 = 31 nM T23995 CGQ7F8 53473746 IC50 = 2.9 nM T23995 CI1ZG3 53473747 IC50 = 0.6 nM T23995 C67JHW 53473748 IC50 = 1.2 nM T23995 C7EW6O 53473749 IC50 = 5.1 nM T23995 CPH34R 53473750 IC50 = 71 nM T23995 CWH1D4 53473825 IC50 > 316 nM T23995 CM8K2V 53473826 IC50 = 7.8 nM T23995 C9A8HG 53473827 IC50 = 316 nM T23995 C3A8OT 53473828 IC50 = 67 nM T23995 CLX31Q 53473829 IC50 = 221 nM T23995 C8Y9RE 53473918 IC50 = 8.3 nM T23995 C1XFN0 53473919 IC50 = 9.8 nM T23995 CN34UO 53473920 IC50 = 7 nM T23995 C2RE5M 53473921 IC50 = 0.1 nM T23995 C9ZUL0 53473922 IC50 = 5.8 nM T23995 CG6FD5 53474007 IC50 = 3.8 nM T23995 C0Q7JS 53474008 IC50 = 26 nM T23995 C31WZB 53474009 IC50 = 1.2 nM T23995 CJF1M2 53630890 IC50 = 263 nM T23995 C1XS2J 54760383 IC50 = 3600 nM T23995 CNB76L 56643505 IC50 = 55 nM T23995 CE25GK 57392822 EC50 = 7140 nM T23995 CB4LH7 57690468 Ki = 6 nM T23995 CG1V8H 57690486 Ki = 275 nM T23995 CP0L8E 57690510 Ki = 20 nM T23995 CS9E2N 57690531 Ki = 7 nM T23995 C2J9WL 57690545 Ki = 0.6 nM T23995 CSG48Q 57690557 Ki = 1975 nM T23995 C6G3FO 57690592 Ki = 1520 nM T23995 CQ4ZT0 57690683 Ki = 238 nM T23995 C4PQX2 57690725 Ki = 38 nM T23995 C4RDK5 57690748 Ki = 375 nM T23995 CEX2M9 57690785 Ki > 2800 nM T23995 CX61LY 57690790 Ki = 76 nM T23995 CQ0OR2 57690846 Ki = 32 nM T23995 CSP2I8 57690850 Ki > 700 nM T23995 CQ9E6Z 57969591 Ki = 5 nM T23995 CAU57Q 57969602 Ki = 2 nM T23995 CHZ4R7 57969605 Ki < 1 nM T23995 C6JNW8 57969629 Ki = 14 nM T23995 CW0BD8 57969638 Ki = 72 nM T23995 C9BY8O 57969654 Ki = 12 nM T23995 C8N7KT 57969691 Ki = 32 nM T23995 C1LZI4 57969746 Ki = 6 nM T23995 CQ30ER 57969765 Ki = 0.2 nM T23995 C7DGA0 57969770 Ki = 0.4 nM T23995 CF7H2Z 57969835 Ki = 30 nM T23995 C0AIT3 58324717 IC50 = 1.3 nM T23995 CL5NT8 58324719 IC50 = 5.4 nM T23995 C5L3OP 58324754 IC50 = 170 nM T23995 CP2YV0 58324879 IC50 = 100 nM T23995 CTS35O 58324901 IC50 = 33 nM T23995 CFQK52 58324920 IC50 = 5.4 nM T23995 C7TJ1A 58324948 IC50 = 60 nM T23995 C24GYC 58325034 IC50 = 28 nM T23995 CPDJ06 58325113 IC50 = 2.7 nM T23995 C9ZQ4A 58325139 IC50 = 1.9 nM T23995 CDJ9R8 58325148 IC50 = 6.4 nM T23995 CT0W2I 58325197 IC50 = 3.1 nM T23995 CA1UT9 58325275 IC50 = 5.2 nM T23995 COH41P 58325285 IC50 = 0.7 nM T23995 C8I6QZ 58325298 IC50 = 39 nM T23995 C50GIS 58325302 IC50 = 130 nM T23995 CA4MI1 58325385 IC50 = 5.9 nM T23995 CU38PN 58367655 Ki = 24 nM T23995 CT3EW2 59292007 IC50 = 320 nM T23995 CJ6ZT2 59332810 IC50 = 496 nM T23995 CXJ63M 59603829 IC50 > 100000 nM T23995 CQEU96 59603842 IC50 = 270 nM T23995 COH62U 60097413 IC50 > 10000 nM T23995 C1MR8Q 60097495 IC50 > 10000 nM T23995 CNL04P 60155126 Ki = 2.9 nM T23995 C56PUM 60155209 Ki = 0.54 nM T23995 CK6WO0 66552478 IC50 < 10000 nM T23995 C1HSE0 67035086 IC50 = 230 nM T23995 CWI6K5 67035106 IC50 > 10000 nM T23995 C37NKO 67129970 IC50 > 10000 nM T23995 CK80LJ 67130050 IC50 > 10000 nM T23995 CV63UL 67240318 IC50 > 10000 nM T23995 CSTC21 67739234 Ki = 745 nM T23995 CVJ2P6 67739562 Ki = 1010 nM T23995 CJM08K 67949700 Ki = 4 nM T23995 CJX61W 67949768 Ki > 700 nM T23995 C2PWR3 67949769 Ki = 5 nM T23995 CJ1CK8 67949771 Ki = 51 nM T23995 CA43IM 67949780 Ki = 9 nM T23995 CWZ6B3 67949822 Ki = 5 nM T23995 C8KR4F 67949825 Ki = 10 nM T23995 C8I7GC 68293638 IC50 > 10000 nM T23995 CD56XK 68293660 IC50 > 10000 nM T23995 CF39DV 68596931 IC50 = 132 nM T23995 C9XLB3 68597337 IC50 = 77 nM T23995 CMQ58W 68597501 IC50 = 743 nM T23995 CEZU83 68611347 IC50 = 948 nM T23995 CLB0J1 68665038 IC50 = 1.5 nM T23995 CJ8G3H 68682755 IC50 > 316 nM T23995 C7GRV2 68755406 IC50 > 10000 nM T23995 C5DGR9 69036886 IC50 = 10000 nM T23995 CJGH31 70285522 IC50 > 1000 nM T23995 CPZ4F6 71451107 IC50 > 1000 nM T23995 C5RKX0 71452928 IC50 > 1000 nM T23995 CEBO91 71452977 IC50 > 10000 nM T23995 CLZ67D 71456431 IC50 > 1000 nM T23995 CS89CL 71456432 IC50 = 350 nM T23995 CHQZ25 71459584 IC50 > 10000 nM T23995 CPIH21 71460129 IC50 = 93 nM T23995 C69NCX 71461845 IC50 > 1000 nM T23995 C9QB5V 71461846 IC50 > 1000 nM T23995 C6O8KG 71461847 IC50 = 738 nM T23995 C07RPM 71583135 Ki = 0.2 nM T23995 C97WFL 71583136 Ki = 133 nM T23995 C07HUA 71583137 Ki = 1 nM T23995 CR2P7K 71583245 Ki = 21 nM T23995 CIQK36 71583246 Ki = 21 nM T23995 C4MOE6 71583247 Ki = 20 nM T23995 CZ31PU 71583657 IC50 > 10000 nM T23995 CV70GZ 71728100 Ki = 0.2 nM T23995 C8Y2HG 75164988 IC50 = 0.7 nM T23995 C4OAP2 76285721 IC50 = 59 nM T23995 CFRU64 76285722 IC50 = 23 nM T23995 CFNV06 76285723 IC50 = 57 nM T23995 CBA6J9 76285725 IC50 = 52 nM T23995 CU80OY 76286333 IC50 = 100 nM T23995 C28COI 76286478 IC50 = 4 nM T23995 C7Q0AD 76286479 IC50 = 49 nM T23995 CZF0N7 76287389 IC50 = 49 nM T23995 C28STM 76287526 IC50 = 55 nM T23995 CON05R 76760640 IC50 < 1 nM T23995 CXSJ93 76760656 IC50 = 0.1 nM T23995 CC0V7I 76760702 IC50 = 43 nM T23995 C25CXS 76760724 IC50 = 0.38 nM T23995 C0IZ5K 76760742 IC50 = 0.42 nM T23995 CG8P0V 76760765 IC50 = 1.4 nM T23995 CSYL29 76760767 IC50 = 0.44 nM T23995 C1CY2S 76760769 IC50 = 1.9 nM T23995 CHW65O 76760780 IC50 = 32 nM T23995 CZB02Q 76760810 IC50 = 0.23 nM T23995 C8JOP4 76760813 IC50 = 0.46 nM T23995 CC3LB6 76760857 IC50 = 18 nM T23995 CMV8Z9 76760918 IC50 = 0.94 nM T23995 C2IK0Z 76760989 IC50 = 140 nM T23995 C0J2OC 76761020 IC50 < 1 nM T23995 COV3R4 76761099 IC50 = 17 nM T23995 CSV23A 78673872 IC50 = 995 nM T23995 C1T9SW 86727297 IC50 = 760 nM T23995 CFB65P 86727308 IC50 = 320 nM T23995 C2L4TA 86727318 IC50 = 390 nM T23995 C3IHT7 86727428 IC50 = 59 nM T23995 CQ6BO2 86727508 IC50 = 3 nM T23995 CL03AB 86727576 IC50 = 4 nM T23995 C06XHV 86727577 IC50 = 3 nM T23995 CCQO02 86727584 IC50 = 16 nM T23995 CNIR39 86727592 IC50 = 43 nM T23995 CC7T6X 86727607 IC50 = 2 nM T23995 C1HW4B 89735655 IC50 = 8700 nM T23995 CM58JI 90219582 IC50 = 2 nM T23995 CNK87H 90219670 IC50 = 110 nM T23995 C2TW8U 90219704 IC50 = 67 nM T23995 CGM7O0 90220574 IC50 = 130 nM T23995 CSO9Z4 90220754 IC50 = 7 nM T23995 CJ84EU 90220857 IC50 = 2 nM T23995 C7J2KY 90230692 IC50 = 8 nM T23995 CH0KN5 90230742 IC50 = 41 nM T23995 CUX8F6 90230745 IC50 = 4 nM T23995 CN67RP 91758287 IC50 = 785 nM T23995 C0Y8ZK 91933875 IC50 = 0.25 nM T23995 CN8A6F 118409668 IC50 = 0.46 nM T23995 C7ZL3Q 118715599 IC50 = 1531 nM T23995 C8T0AY 118715600 IC50 > 1000 nM T23995 C2J3YZ 118715601 IC50 > 1000 nM T23995 CRG06J 118715602 IC50 > 1000 nM T23995 C7WS3V 118715603 IC50 > 1000 nM T23995 CQM81J 118715604 IC50 > 1000 nM T23995 C7FM1Z 118720640 IC50 = 700 nM T23995 CXM16L 118720641 IC50 = 42 nM T23995 CH8QZ0 118720642 IC50 = 3 nM T23995 CAL3R5 118720643 IC50 = 5 nM T23995 CT73PB 118720644 IC50 = 14 nM T23995 CRQ30U 118720645 IC50 = 19 nM T23995 C0T3PE 118720646 IC50 = 24 nM T23995 CS41FQ 118720647 IC50 = 10 nM T23995 CESF83 118720648 IC50 = 240 nM T23995 CHS2B7 118720649 IC50 = 5 nM T23995 CJV1D9 118720650 IC50 = 190 nM T23995 CTG46P 118721283 IC50 = 16000 nM T23995 CTK8O0 118721284 IC50 = 1300 nM T23995 CGE75Y 118721285 IC50 = 38000 nM T23995 CRQ07H 118721545 IC50 > 50000 nM T23995 CH35QW 118721546 IC50 = 3300 nM T23995 C3OM6T 118721547 IC50 = 14000 nM T23995 CH8VT7 118721548 IC50 = 21000 nM T23995 CAR0E9 118721549 IC50 = 8900 nM T23995 C5U9NA 118721550 IC50 = 17000 nM T23995 C4A9NT 118721551 IC50 = 20000 nM T23995 CHTM28 118721552 IC50 = 31000 nM T23995 C69NJC 118721553 IC50 = 18000 nM T23995 CW17XA 118721554 IC50 = 46000 nM T23995 C4MTN3 118721555 IC50 = 19000 nM T23995 CB43SF 118721556 IC50 = 46000 nM T23995 CDK37Z 118721557 IC50 = 3500 nM T23995 CJF2O4 118721558 IC50 = 4500 nM T23995 C6WBM0 118721559 IC50 > 50000 nM T23995 CYK02G 118721560 IC50 = 230 nM T23995 CDL8V3 118721561 IC50 = 1000 nM T23995 CTS0Y7 118721562 IC50 = 3500 nM T23995 C58EWT 118721563 IC50 > 50000 nM T23995 CV4O8P 118721564 IC50 = 190 nM T23995 CZ98MP 122180028 IC50 = 4 nM T23995 CTR5Y6 122180029 IC50 = 0.68 nM T23995 CE54RP 122180030 IC50 = 5.2 nM T23995 CG06LU 122180031 IC50 = 0.32 nM T23995 C9D4PT 122180032 IC50 = 0.14 nM T23995 C0HQB2 122180033 IC50 = 0.46 nM T23995 CWUR30 122180034 IC50 = 30 nM T23995 CA8B4N 122180035 IC50 > 100 nM T23995 C9VRW7 122180036 IC50 = 2.1 nM T23995 C4SXY8 122180037 IC50 = 10 nM T23995 C6OS9Y 122180038 IC50 = 27 nM T23995 C0B2IO 122180039 IC50 = 28 nM T23995 CUWZ20 122180040 IC50 = 32 nM T23995 CQ9OW0 122180041 IC50 = 3 nM T23995 C38HIM 127046041 IC50 = 170 nM T23995 CMGE71 127046440 IC50 = 260 nM T23995 CX2ND0 127047219 IC50 = 60 nM T23995 C3YIJ8 127047265 IC50 = 45 nM T23995 CCB84X 127047266 IC50 = 12 nM T23995 C7JH3L 127047340 IC50 = 300 nM T23995 CJ5G3I 127047392 IC50 = 170 nM T23995 CV5PJ1 127047393 IC50 = 150 nM T23995 CK8XV0 127047535 IC50 = 100 nM T23995 CRX9A2 127048046 IC50 = 930 nM T23995 CRSW19 127048047 IC50 = 240 nM T23995 CI5AM0 127048048 IC50 = 1900 nM T23995 C8F0DQ 129909860 IC50 = 7 nM T23995 CSB0M9 135494223 EC50 = 7250 nM T23995 CEK31P 135566415 IC50 > 20000 nM T23995 CX4ZB3 135863110 IC50 = 25900 nM T23995 C1XQY2 135923992 EC50 = 3160 nM T23995 CC65KF 136042192 EC50 = 15840 nM T23995 CZ7EX0 136183413 IC50 = 22400 nM T23995 CJ7KN6 136250327 Ki = 0.1 nM T23995 C31DIA 137633180 IC50 = 0.18 nM T23995 CI1E8V 137634241 IC50 > 10000 nM T23995 CG0WZ8 137634847 IC50 = 250 nM T23995 CG8M4U 137638978 IC50 = 100 nM T23995 C12UXT 137640959 IC50 > 316 nM T23995 CH15QZ 137643717 IC50 = 254 nM T23995 C84EOJ 137646250 IC50 = 0.086 nM T23995 C73XQU 137647557 IC50 > 1000 nM T23995 C8LE6Y 137651788 IC50 = 18 nM T23995 C12LWY 137654723 IC50 = 6.7 nM T23995 CWPJ25 137655826 IC50 = 0.87 nM T23995 C2QX6B 137659527 IC50 = 14 nM T23995 CUG6N7 137660315 IC50 = 21 nM T23995 CYC5U2 137660537 IC50 = 33 nM T23995 C6S5FI 137660962 IC50 = 6.3 nM T23995 C6QA5D 137661222 IC50 > 316 nM T23995 C7I3UR 145979852 IC50 = 51 nM T23995 C7XU0Q 145980343 IC50 = 24 nM T23995 C2YK4I 145981931 IC50 = 36 nM T23995 CL95US 145989117 IC50 = 130 nM T23995 CAZ94J 145991320 IC50 = 14 nM T23995 CQA1I3 145993975 IC50 = 4.6 nM T23995 C2MD1Q 155513187 IC50 > 10000 nM T23995 CPA8W3 155519578 IC50 > 100 nM T23995 CU34OH 155567589 Ki = 8 nM T23995 D02KPV 37783 Ki = 1.54 nM T23995 D04AXH 11574614 Ki = 290 nM T23995 D06HVH 54613583 IC50 = 1400 nM T23995 D07ANB 148879 EC50 = 5240 nM T23995 D08HCY 45485036 IC50 = 1400 nM T23995 D0K5ZY 105000 Ki = 8.7 nM T23995 D0S7UD 45484993 IC50 = 690 nM T23995 D0TO6S 2396 IC50 = 6.7 nM T23995 D0U9YY 45485012 IC50 = 24 nM T06850 D0W9VW 11526696 Ki = 16 nM T06850 C7HNP0 11526745 Ki = 2.6 nM T06850 CG0WP3 11541143 Ki = 34 nM T06850 C9F5DJ 11541319 Ki = 61 nM T06850 C9MOG2 11664206 Ki = 7 nM T06850 C56FEK 11692516 Ki = 15 nM T06850 C7VNL2 11706547 Ki = 104 nM T06850 CK04CH 24969520 Ki = 34 nM T06850 CFHG08 24969603 Ki = 5 nM T06850 CG9B3J 24970113 Ki = 0.38 nM T06850 CP78UW 56925343 Ki = 0.9 nM T06850 CY83AU 56925344 Ki = 19 nM T06850 C6Q8KJ 56925345 Ki = 58 nM T06850 CP1W5M 56926173 Ki = 86 nM T06850 CI56WR 56926174 Ki > 10000 nM T06850 CTY13B 56926175 Ki = 68 nM T06850 C1GE5S 56926176 Ki = 1200 nM T06850 CZO13G 56926177 Ki = 380 nM T06850 C3XME7 56926265 Ki > 10000 nM T06850 C2WK6M 56926266 Ki = 1100 nM T06850 C31DMQ 56926267 Ki > 10000 nM T06850 C4K5VS 56926268 Ki = 670 nM T06850 C0NZM5 56926269 Ki = 400 nM T06850 C7LR2A 56926356 EC50 = 39 nM T06850 CLV81C 56926357 Ki > 10000 nM T06850 CZ6UI4 56926358 Ki > 10000 nM T06850 C3WNX0 56926359 Ki > 10000 nM T06850 CNWF73 56926360 Ki = 25 nM T06850 C30RQU 56926461 Ki = 6.4 nM T06850 CP9I4G 56926462 Ki = 4.4 nM T06850 C4EM7N 56926463 Ki = 16 nM T06850 C97NEM 56926464 Ki = 580 nM T06850 CV6XU4 56926465 Ki = 500 nM T06850 CQ45BS 56926580 Ki = 35 nM T06850 C16OSK 56926581 Ki = 380 nM T06850 C0VY2C 56926582 Ki = 43 nM T06850 CIN53V 56926584 Ki = 32 nM T06850 CQX09U 56926680 Ki = 6.2 nM T06850 C09URY 56926681 Ki = 21 nM T06850 C2DP7T 56926682 Ki = 7.3 nM T06850 C4Z6CM 56926781 Ki > 10000 nM T06850 CSI61U 56926782 Ki = 1500 nM T06850 CP28XJ 56926783 Ki = 160 nM T06850 CYP26U 56926784 Ki = 400 nM T06850 CHS0A1 56926785 Ki = 210 nM T06850 CQ4G5W 56926891 Ki = 81 nM T06850 CXR9Q6 56926892 Ki = 78 nM T06850 CF0KR5 56926893 Ki = 9 nM T06850 CGU3Q4 56926894 EC50 = 26 nM T06850 CG3RD4 56926895 Ki = 12 nM T06850 CTC13B 57390496 Ki = 4.8 nM T06850 C8CG2S 57399248 Ki = 0.35 nM T31621 CGP74I 10485791 IC50 = 20000 nM T31621 C1E2SY 44340157 IC50 = 0.01 ug.mL-1 T31621 CRW4A6 44340520 IC50 = 0.058 ug.mL-1 T31621 CCG32P 44340522 IC50 = 11 ug.mL-1 T31621 CS40UM 71718463 IC50 < 0.1 ug.mL-1 T31621 CUN1B2 97290924 IC50 = 10000 nM T31621 CS2T8P 127053051 IC50 = 10000 nM T31621 C4V2NK 145965586 IC50 = 271000 nM T31621 C6SU5D 145977503 IC50 = 42000 nM T31621 C1K0TP 154702460 IC50 = 1300 nM T54065 CYK45N 8742 IC50 > 90000000 nM T54065 CM92TF 41910 Ki = 2200 nM T54065 CCF9V8 132878 Ki = 7400 nM T54065 CMZP14 192265 Ki = 85000 nM T54065 C6HI1T 349158 IC50 = 50000000 nM T54065 C0KF3T 541499 Ki = 78000 nM T54065 CKB06Y 808704 Ki = 650 nM T54065 CVM30A 5289341 Ki 0.11 nM T54065 C2R5WQ 9990447 IC50 = 50000000 nM T54065 CVG45E 12795583 IC50 > 1000 nM T54065 CJ5IO7 12832584 IC50 > 80000 nM T54065 CJ4YV7 13021075 Ki = 2200 nM T54065 CW02LT 13512182 IC50 = 700000 nM T54065 C3MVX5 15059815 Ki = 13000 nM T54065 C7MYI6 15747604 Ki = 1500 nM T54065 CFI98B 20697688 IC50 = 15000000 nM T54065 CQXJ83 20697689 IC50 > 90000000 nM T54065 CZ0PE9 44281432 IC50 > 90000000 nM T54065 C7BJ1N 44281433 IC50 = 7500000 nM T54065 CJA2G8 44281440 IC50 > 90000000 nM T54065 C0J4FD 44281442 Ki = 1500 nM T54065 CZGE84 44281452 IC50 > 90000000 nM T54065 C0USA5 44281473 IC50 > 90000000 nM T54065 CZ7D0P 44281691 IC50 > 90000000 nM T54065 CCV4H1 44281693 IC50 > 90000000 nM T54065 CVUD18 44281694 IC50 > 90000000 nM T54065 C7N1YZ 44281708 IC50 = 180000 nM T54065 C1KX2O 44321575 Ki = 780 nM T54065 CP8Z9A 44321577 IC50 = 10000000 nM T54065 CGCV15 44321833 IC50 = 1400000 nM T54065 C4WJB5 44321835 IC50 = 10000000 nM T54065 CW68CR 44321836 IC50 = 10000000 nM T54065 C4FDS9 44321837 Ki = 2500 nM T54065 CN6U0M 44321861 Ki = 1500 nM T54065 CWMQ01 44321865 IC50 = 3000000 nM T54065 CI4RL3 44321873 IC50 > 80000000 nM T54065 CX10EA 44321919 Ki = 160 nM T54065 C1BJP5 44328529 IC50 = 50000000 nM T54065 CVY6P4 44328660 Ki = 1300 nM T54065 CR1O4X 44328706 Ki = 520 nM T54065 CWGU46 44328787 IC50 = 20000000 nM T54065 CH2NJ3 44328832 IC50 > 10000000 nM T54065 CB59HP 44328952 Ki = 5200 nM T54065 C7QX1P 44329017 IC50 > 80000 nM T54065 C4O7GC 44329285 IC50 > 80000 nM T54065 C6J9RK 44329294 Ki = 610 nM T54065 CZ5T8D 44356177 Ki = 100 nM T54065 C9G1VQ 53317222 IC50 = 2000000 nM T54065 C97BYX 53318522 Ki = 5 nM T54065 CH62GC 53321137 IC50 = 10000000 nM T54065 C7CY1I 53321139 Ki = 160 nM T54065 CZRK61 53322470 Ki = 4 nM T54065 C4A0TX 53323824 IC50 = 7900000 nM T54065 CD8G1Q 53326392 Ki = 32 nM T54065 C1QI4G 54733255 IC50 = 7900000 nM T54065 D04HMD 3496 Ki = 160 nM T83391 D06ACW 6083 IC50 = 140 nM T83391 D0Q7HO 4705 IC50 = 1000 nM T83391 CH21PG 2428 IC50 = 4000 nM T83391 CGZ59Q 65110 IC50 = 12000 nM T83391 CB4K2F 211386 IC50 = 320180 nM T83391 CC1V0H 446916 IC50 = 2000 nM T83391 C8J1FN 819894 IC50 = 490 nM T83391 CNIE06 5284459 IC50 = 3500 nM T83391 CB35RO 5328213 IC50 = 11900 nM T83391 C1SR4I 5328218 IC50 > 10000 nM T83391 CQ3MT4 5328219 IC50 > 10000 nM T83391 CIEL17 5328225 IC50 = 4500 nM T83391 CFW19M 5329009 IC50 = 290 nM T83391 C8JQI5 5702506 IC50 = 1100 nM T83391 CXB7A0 6102820 IC50 = 3400 nM T83391 CBP16R 6102822 IC50 = 570 nM T83391 CQZ1J8 9798527 IC50 = 800 nM T83391 CJV87E 9811837 IC50 = 10 nM T83391 CG5L7Z 9842886 IC50 = 55 nM T83391 C2DL8U 9927208 IC50 = 250 nM T83391 CW5U1T 10048580 IC50 = 2100 nM T83391 C8Q9XW 10451264 IC50 = 530 nM T83391 CR8XL6 10895415 IC50 > 10000 nM T83391 CPB40Z 11123661 IC50 > 10000 nM T83391 C5KI6F 11134028 IC50 > 10000 nM T83391 C6C1EU 11289630 EC50 = 16 nM T83391 CZ2E6X 11660897 IC50 = 1600 nM T83391 CH6J9V 11710304 IC50 = 9200 nM T83391 C57MTX 11949961 IC50 = 15 nM T83391 C60MXV 11949964 IC50 = 2 nM T83391 CM7W8T 11950133 IC50 = 11 nM T83391 C4QL0Y 11950134 IC50 = 10 nM T83391 C5W7AX 12037178 IC50 = 1400 nM T83391 C7T3HI 14177233 IC50 = 12700 nM T83391 CRQ1G5 15895242 IC50 = 2250 nM T83391 C6V5EB 15895245 IC50 = 6000 nM T83391 C8X4RP 15950347 IC50 = 2500 nM T83391 C3ZC6E 16045442 IC50 = 900 nM T83391 CN63KT 16079088 IC50 = 1 nM T83391 CA7C0Y 18925067 IC50 = 2400 nM T83391 CV3FQ7 20737671 IC50 = 120 nM T83391 CU8VJ7 20737672 IC50 = 16 nM T83391 C2VM4Z 22280501 IC50 = 50 nM T83391 CER74G 22280522 IC50 = 380 nM T83391 CBOR90 22280555 IC50 = 350 nM T83391 C0SPR1 22280574 IC50 = 420 nM T83391 CC9TB3 22280600 IC50 = 250 nM T83391 C7ZDX3 22280622 IC50 = 7000 nM T83391 CQL0O9 22280633 IC50 = 950 nM T83391 C5F1NQ 22280709 IC50 = 55 nM T83391 CX4T8E 22280713 IC50 = 580 nM T83391 C6MPW2 22280715 IC50 = 280 nM T83391 C03JUW 22321091 IC50 = 2500 nM T83391 CW7EP1 22321151 IC50 = 100 nM T83391 CNT34U 22459816 IC50 = 60 nM T83391 CYNS79 22459821 IC50 = 3000 nM T83391 CZ8CA4 22459827 IC50 = 500 nM T83391 C31EXG 22459828 IC50 = 130 nM T83391 C5T9ZB 22459832 IC50 = 90 nM T83391 C6MDJ5 22459834 IC50 = 80 nM T83391 C6T0CS 22459869 IC50 = 100 nM T83391 C1BWF9 22459880 IC50 = 700 nM T83391 C91ELW 22459908 IC50 = 280 nM T83391 C56TZE 22459919 IC50 = 450 nM T83391 CG0K6L 22459920 IC50 = 90 nM T83391 C6CBD9 22459922 IC50 = 225 nM T83391 CGLF84 22459925 IC50 = 70 nM T83391 CHO1X7 22459931 IC50 = 100 nM T83391 CBJQ54 22459932 IC50 = 180 nM T83391 CC3FU1 22459935 IC50 = 150 nM T83391 CDLQ13 23103191 IC50 = 600 nM T83391 C32LKB 23733120 IC50 = 6200 nM T83391 CC36EV 24751654 IC50 = 140 nM T83391 C57NUW 24751659 IC50 = 190 nM T83391 C5T4JW 24751933 IC50 = 380 nM T83391 CM54YI 24751937 IC50 = 380 nM T83391 C7P8WL 24752079 IC50 = 90 nM T83391 C6R2DP 24752215 IC50 = 100 nM T83391 CFIK61 24752216 IC50 = 290 nM T83391 CADB19 24752360 IC50 = 100 nM T83391 CXS03C 24752361 IC50 = 80 nM T83391 C53RPX 24752501 IC50 = 170 nM T83391 C20WPN 24752505 IC50 = 90 nM T83391 C9UP1L 24752506 IC50 = 60 nM T83391 C9RA5C 24752507 IC50 = 40 nM T83391 CI8SX5 24752643 IC50 = 40 nM T83391 CCF16E 24752645 IC50 = 70 nM T83391 C7XFB1 24752646 IC50 = 320 nM T83391 C35TAV 24752648 IC50 = 70 nM T83391 CVF9C5 24752786 IC50 = 210 nM T83391 COW34C 24752787 IC50 = 50 nM T83391 CTZ5U2 24752788 IC50 = 120 nM T83391 C51OGU 24752790 IC50 = 170 nM T83391 C5RH3W 24762220 IC50 = 8 nM T83391 CZ4MN8 24780158 IC50 = 330 nM T83391 CUHE51 24780310 IC50 = 30 nM T83391 C5KYL1 24780311 IC50 = 90 nM T83391 CL8QB4 24856345 IC50 = 4 nM T83391 CHAD10 24963320 IC50 = 4 nM T83391 C9M3WI 24963322 IC50 = 2 nM T83391 C1A4QM 24963667 IC50 = 12 nM T83391 CHS9T6 24964016 IC50 = 12 nM T83391 C6WZ0T 24964736 IC50 = 28 nM T83391 C2UX7V 24965099 IC50 = 22 nM T83391 C9LC1B 24965449 IC50 = 35 nM T83391 CWER10 24965450 IC50 = 5 nM T83391 CJ09XT 24968298 IC50 = 17 nM T83391 C30HJP 24968299 IC50 = 19 nM T83391 CJT7C2 24968646 IC50 = 16 nM T83391 CZH0T5 24968648 IC50 = 14 nM T83391 C7Y9ZM 24968649 IC50 = 24 nM T83391 CQUJ60 42628889 IC50 = 520 nM T83391 CSW5D7 42628891 IC50 = 350 nM T83391 C3IB0D 42629276 IC50 = 80 nM T83391 CLX25A 42629393 IC50 = 130 nM T83391 C3X4TP 42629397 IC50 = 170 nM T83391 C04MBY 42629630 IC50 = 400 nM T83391 CH96QK 42629631 IC50 = 1800 nM T83391 C74NWB 42629632 IC50 = 1700 nM T83391 C9A0FC 42630357 IC50 = 600 nM T83391 CF6D1A 42630482 IC50 = 670 nM T83391 CNV2H3 42630485 IC50 = 420 nM T83391 CIRV69 42630486 IC50 = 760 nM T83391 C41CLA 42633650 IC50 = 410 nM T83391 CHNJ06 42634013 IC50 = 80 nM T83391 C1TX5U 42634015 IC50 = 70 nM T83391 C4JU5P 42634696 IC50 = 90 nM T83391 CNO1L3 42635072 IC50 = 390 nM T83391 C68QBS 42635430 IC50 = 70 nM T83391 CE5UH4 42635792 IC50 = 100 nM T83391 C4R0FM 42637217 IC50 = 2000 nM T83391 CG72WI 42637218 IC50 = 1800 nM T83391 CJZY67 42637219 IC50 > 10000 nM T83391 CIQ9A6 42637288 IC50 = 900 nM T83391 CVZ54G 42637289 IC50 = 5000 nM T83391 CR02EU 42637290 IC50 > 10000 nM T83391 C2IKT8 42637292 IC50 = 13000 nM T83391 C09QKC 42637293 IC50 = 5500 nM T83391 CE98LD 42637368 IC50 = 700 nM T83391 CFO0U6 42637645 IC50 > 100000 nM T83391 CG2I7W 42637646 IC50 > 100000 nM T83391 C35HLT 42637647 IC50 = 140000 nM T83391 CJS53Q 42637648 IC50 = 91000 nM T83391 C8QE6L 42637712 IC50 = 100000 nM T83391 C54ORK 42637714 IC50 = 23000 nM T83391 CLJ0D3 42637715 IC50 > 500000 nM T83391 C9SF4V 42637717 IC50 = 100000 nM T83391 CX85JL 42637718 IC50 = 145000 nM T83391 C09KPG 42637779 IC50 > 100000 nM T83391 CKDC59 42637780 IC50 = 48000 nM T83391 CRQ80D 42637783 IC50 = 40000 nM T83391 COJ91B 42637784 IC50 = 150000 nM T83391 CSGL53 42637785 IC50 = 250000 nM T83391 C35MSX 42637843 IC50 = 50000 nM T83391 C50VUA 42637844 IC50 = 3300 nM T83391 CL34WC 42637849 IC50 > 100000 nM T83391 CN43CE 42637919 IC50 = 100000 nM T83391 CQOC90 42637922 IC50 = 35000 nM T83391 C8F0IN 42637923 IC50 = 100000 nM T83391 C7BM2D 42637924 IC50 = 100000 nM T83391 CRY27L 42637925 IC50 > 1000000 nM T83391 C94ETG 42637998 IC50 > 100000 nM T83391 C9U2BI 42637999 IC50 > 100000 nM T83391 C7HV8W 42638000 IC50 = 50000 nM T83391 CN18AQ 42638001 IC50 = 70000 nM T83391 C9D0GV 42638002 IC50 = 1500 nM T83391 CHU07P 42638077 IC50 = 28000 nM T83391 C0EXH7 42638078 IC50 = 4500 nM T83391 C5WD9L 42638079 IC50 = 1600 nM T83391 CYC3F7 42638080 IC50 = 1100 nM T83391 CPXF17 42638082 IC50 > 100000 nM T83391 C4OHG0 44306424 IC50 > 10000 nM T83391 C1H4RI 44306425 IC50 > 10000 nM T83391 C1B0CR 44306428 IC50 > 10000 nM T83391 CGA4D8 44306455 IC50 > 10000 nM T83391 CA5J9L 44306459 IC50 = 5500 nM T83391 C1YXE0 44306472 IC50 = 2900 nM T83391 CUKH60 44306495 IC50 > 10000 nM T83391 C8DNU6 44306496 IC50 > 10000 nM T83391 CCKP73 44306529 IC50 > 10000 nM T83391 CWK5R1 44306530 IC50 > 10000 nM T83391 CSO10Y 44306531 IC50 > 10000 nM T83391 CQIP27 44306541 IC50 > 10000 nM T83391 C2UZL7 44306632 IC50 > 10000 nM T83391 C2UZR7 44306833 IC50 > 10000 nM T83391 CQ2M4I 44306834 IC50 > 10000 nM T83391 C4TJ3C 44306917 IC50 = 3600 nM T83391 CV7T4E 44409652 IC50 > 50000 nM T83391 CA7O2S 44409655 IC50 = 2800 nM T83391 C83JZC 44409656 IC50 = 7800 nM T83391 CM5SL0 44409657 IC50 = 6400 nM T83391 CK1HT0 44409662 IC50 = 32000 nM T83391 C63NPS 44409663 IC50 = 4000 nM T83391 CQYL73 44409668 IC50 = 8100 nM T83391 CR97PD 44409682 IC50 = 10000 nM T83391 C6NBR3 44409792 IC50 = 3400 nM T83391 CE9B2N 44409795 IC50 = 8000 nM T83391 CDO37J 44409798 IC50 = 6000 nM T83391 C41QGF 44409804 IC50 = 3800 nM T83391 C68FCU 44409805 IC50 = 24000 nM T83391 CJS5H3 44409811 IC50 = 4000 nM T83391 CO60MD 44409812 IC50 = 6700 nM T83391 C0BDT5 44409814 IC50 = 12000 nM T83391 CDZ1L2 44409815 IC50 = 2600 nM T83391 C5BU0K 44409822 IC50 = 1300 nM T83391 C75ISX 44409836 IC50 > 50000 nM T83391 CMR35B 44409837 IC50 > 50000 nM T83391 C50JQE 44409838 IC50 = 6500 nM T83391 CVP81Z 44409847 IC50 > 50000 nM T83391 CHAF34 44409848 IC50 > 50000 nM T83391 C84PZA 44409849 IC50 = 6200 nM T83391 C10PZI 44409850 IC50 = 3500 nM T83391 C8MC7K 44409851 IC50 = 1700 nM T83391 CXF53K 44409854 IC50 > 50000 nM T83391 C6GQX1 44409855 IC50 = 1800 nM T83391 CM2RG5 44409972 IC50 = 23000 nM T83391 CI2DF8 44409991 IC50 = 55000 nM T83391 CD3G7L 44409997 IC50 = 1900 nM T83391 CUC37B 44410043 IC50 = 13000 nM T83391 C2VU7P 44410044 IC50 = 9400 nM T83391 C9RYL6 44410048 IC50 = 1300 nM T83391 C7K5OR 44410049 IC50 = 1800 nM T83391 CJR4A0 44410050 IC50 = 9800 nM T83391 C5WX9D 44568648 IC50 = 14 nM T83391 CFHN94 44568649 IC50 = 14 nM T83391 C3KPX2 44587556 IC50 > 100000 nM T83391 C9GW4C 44587558 IC50 = 38530 nM T83391 CJ59VS 44587601 IC50 = 264 nM T83391 C67IGQ 44587602 IC50 = 542 nM T83391 C3MBC1 44587805 IC50 = 18 nM T83391 CD10IH 44587807 IC50 = 151 nM T83391 C9H1KF 44587838 IC50 > 100000 nM T83391 CAJY42 44587839 IC50 = 10 nM T83391 C47JPK 44587840 IC50 = 12 nM T83391 C7NEA4 44587869 IC50 = 57 nM T83391 C94NGZ 44587871 IC50 = 13727 nM T83391 C80ILD 44587904 IC50 = 234231 nM T83391 CD60IB 44587905 IC50 = 134180 nM T83391 CK25HO 44587906 IC50 = 86763 nM T83391 CQK92U 44587909 IC50 = 277143 nM T83391 CA15CZ 44591529 IC50 = 1500 nM T83391 C9NLV5 44591530 IC50 > 10000 nM T83391 CY64EW 44591593 IC50 > 10000 nM T83391 COL7K0 44591594 IC50 > 10000 nM T83391 CSG57B 44591694 IC50 > 100000 nM T83391 CITC73 44591695 IC50 > 100000 nM T83391 C1Z6AY 44591721 IC50 = 100000 nM T83391 CH7I3A 44591722 IC50 > 100000 nM T83391 CLQ47H 44591723 IC50 > 100000 nM T83391 CN5GL0 44591776 IC50 = 5000 nM T83391 CKF3D1 44591798 IC50 > 1000000 nM T83391 C3EQ7H 44591799 IC50 > 1000000 nM T83391 CIV68F 44591800 IC50 > 1000000 nM T83391 CY5F0U 44610740 IC50 = 13 nM T83391 CV18CW 44610756 IC50 = 47 nM T83391 C4DM6S 44626750 IC50 = 1100 nM T83391 COLQ47 44626751 IC50 = 800 nM T83391 CJ2CV5 44626752 IC50 = 800 nM T83391 CNU7X9 44626753 IC50 = 1500 nM T83391 CUEJ29 44626754 IC50 = 2500 nM T83391 CB3F4I 44626755 IC50 = 3250 nM T83391 CT2XY8 44626845 IC50 = 5000 nM T83391 CX90SE 44626846 IC50 = 9500 nM T83391 CJSA81 44626847 IC50 = 7000 nM T83391 C3BTR7 44626848 IC50 = 2500 nM T83391 CZ7G5F 44626849 IC50 = 4200 nM T83391 C5HEF6 44626850 IC50 = 1850 nM T83391 CK92AT 44626939 IC50 = 4000 nM T83391 C1LT6F 44627038 IC50 = 200 nM T83391 CJW15P 44627039 IC50 = 900 nM T83391 CF04RD 44627137 IC50 = 400 nM T83391 CZO32L 44627138 IC50 = 400 nM T83391 CWE1D3 44627139 IC50 = 850 nM T83391 C0Y4JF 44627140 IC50 = 1000 nM T83391 CE52AO 44627250 IC50 = 10000 nM T83391 CI8Z6K 44627368 IC50 = 100 nM T83391 C5PZ1C 44627369 IC50 = 210 nM T83391 C6LKR0 44627481 IC50 = 55 nM T83391 CRCY35 45487191 IC50 = 1000 nM T83391 C8FX3U 45487213 IC50 = 1500 nM T83391 CC3NG0 45487787 IC50 = 19100 nM T83391 C9BF0A 45487792 IC50 = 21500 nM T83391 C7PM4F 45487793 IC50 = 41700 nM T83391 COR31V 45487794 IC50 = 840 nM T83391 C3PX0G 45487808 IC50 = 335000 nM T83391 CD64FS 45487810 IC50 = 22 nM T83391 CY26ZT 45487811 IC50 = 91900 nM T83391 C1XMS6 45487812 IC50 = 18700 nM T83391 CH8MI4 45487818 IC50 = 28400 nM T83391 CL84IN 45487819 IC50 = 354000 nM T83391 C5IT7O 45487820 IC50 = 9320 nM T83391 CZQ3O4 45487822 IC50 = 354000 nM T83391 C7IWP0 45487823 IC50 = 169 nM T83391 C74KLS 45487824 IC50 = 146000 nM T83391 C65TXV 45487827 IC50 = 307000 nM T83391 C93VQI 45487828 IC50 = 70 nM T83391 C7YF1G 45487829 IC50 = 112000 nM T83391 CNGH36 45487833 IC50 = 112000 nM T83391 C59ZXM 45487847 IC50 = 112000 nM T83391 C4H3TO 45487848 IC50 = 124 nM T83391 C8T5MO 45487849 IC50 = 16400 nM T83391 CU19QN 46193619 IC50 = 8100 nM T83391 CS96AK 46193620 IC50 = 6000 nM T83391 C9UD0I 46216773 IC50 = 12 nM T83391 C7OLI2 46224737 IC50 = 310 nM T83391 CP92YX 46224738 IC50 = 530 nM T83391 C74DZU 46224826 IC50 = 180 nM T83391 CS98IR 46224868 IC50 = 180 nM T83391 C38AZF 46224869 IC50 = 260 nM T83391 COJ1U7 46224902 IC50 = 300 nM T83391 CJNZ54 46224903 IC50 = 40 nM T83391 CCV93M 46224904 IC50 > 100000 nM T83391 C3RG8J 46224905 IC50 > 100000 nM T83391 C60KXF 46225257 IC50 = 3500 nM T83391 CGC5R3 46225258 IC50 = 720 nM T83391 C10IRW 46231156 IC50 = 995 nM T83391 CV02MO 46231157 IC50 = 908 nM T83391 C3JV6Q 46231158 IC50 = 772 nM T83391 CNQA41 46231159 IC50 = 8 nM T83391 CVD75O 46231211 IC50 = 8 nM T83391 C1QP7A 46231212 IC50 = 9 nM T83391 CUB38T 46231213 IC50 = 28 nM T83391 C6DWF8 46231214 IC50 = 40 nM T83391 C8ZX5W 46231259 IC50 = 9 nM T83391 C8C7SP 46231260 IC50 = 9 nM T83391 CW21SA 46231261 IC50 = 3 nM T83391 CNIH96 46888798 IC50 = 10 nM T83391 CLKP15 49799630 IC50 = 1 nM T83391 C4LC7B 49799631 IC50 = 2 nM T83391 CU1M6V 49799635 IC50 = 11 nM T83391 C79RCM 49799636 IC50 = 8 nM T83391 C5Q4FE 49799637 IC50 = 11 nM T83391 C5MEJ6 49799646 IC50 = 10 nM T83391 CJR3I8 49799647 IC50 = 10 nM T83391 C73RSF 50992507 IC50 = 300 nM T83391 C0OU6J 50992508 IC50 = 1700 nM T83391 C75WDE 50992509 IC50 = 15 nM T83391 CV39EG 50992510 IC50 = 858 nM T83391 CJQ5H0 50992511 IC50 = 43 nM T83391 C9Y5QN 50992512 IC50 = 21 nM T83391 CF0A1O 50992513 IC50 = 22 nM T83391 C4X1OW 50992514 IC50 = 21 nM T83391 CU49NT 50992584 IC50 = 88 nM T83391 C2R9UK 50992585 IC50 = 14 nM T83391 C3Y1NA 50992586 IC50 = 16 nM T83391 C86ZFB 50992587 IC50 = 13 nM T83391 CWGZ54 50992588 IC50 = 32 nM T83391 CD84FU 50992589 IC50 = 41 nM T83391 CNFS91 50992590 IC50 = 34 nM T83391 C7O9MA 50992649 IC50 = 12 nM T83391 C21OAF 50992650 IC50 = 40 nM T83391 CE86NA 50992651 IC50 = 44 nM T83391 C58FHQ 50992653 IC50 = 10000 nM T83391 CWH8U5 50992654 IC50 = 2000 nM T83391 C5OS3P 50992655 IC50 = 1300 nM T83391 CYFH58 50992729 IC50 = 250 nM T83391 CAJQ97 50992872 IC50 = 24 nM T83391 CJ6A7I 50992874 IC50 = 560 nM T83391 CR8Y5X 50993358 IC50 = 100 nM T83391 CF31ZN 50993359 IC50 = 400 nM T83391 COX93I 50993360 IC50 = 1200 nM T83391 CY1AW3 50993361 IC50 = 220 nM T83391 CQ81LC 50993362 IC50 = 180 nM T83391 CC7EJ5 50993363 IC50 = 80 nM T83391 C6A0JU 50993364 IC50 = 890 nM T83391 CRZO92 50993365 IC50 = 2000 nM T83391 C1YP8I 50993366 IC50 = 1000 nM T83391 C8A3TZ 50993442 IC50 = 10000 nM T83391 C6H7IW 50993443 IC50 = 2750 nM T83391 C04NVS 50993444 IC50 = 500 nM T83391 C1TZ4O 50993445 IC50 = 13500 nM T83391 C0FSV3 50993446 IC50 = 8000 nM T83391 C4J7TI 50993447 IC50 = 5000 nM T83391 C90ZEM 50993448 IC50 = 120 nM T83391 C8TED3 50993449 IC50 = 28 nM T83391 CS7D2K 50993522 IC50 = 57 nM T83391 CQI68N 50993523 IC50 = 12 nM T83391 CCM5N4 50993524 IC50 = 19 nM T83391 C1F4TB 50993525 IC50 = 21 nM T83391 C5CY6B 50993526 IC50 = 10 nM T83391 C9KI6J 50993527 IC50 = 20 nM T83391 CG8O6F 50993528 IC50 = 18 nM T83391 C9OQ1M 50993529 IC50 = 59 nM T83391 CQ81YF 50993601 IC50 = 150 nM T83391 C1BN9K 50993602 IC50 = 70 nM T83391 CP8LZ7 50993603 IC50 = 50 nM T83391 C1C2SE 50993604 IC50 = 100 nM T83391 COW1R5 50993605 IC50 = 16 nM T83391 C4O5CW 50993606 IC50 = 33 nM T83391 CO60JC 50993607 IC50 = 24 nM T83391 C35MQH 51371083 IC50 = 220 nM T83391 C58YKW 53235502 IC50 = 530 nM T83391 CIU0Z4 53316654 IC50 = 135 nM T83391 C1V6UX 53319305 IC50 = 210 nM T83391 CKCO62 53319306 IC50 = 80 nM T83391 CWRJ12 53319346 IC50 > 10000 nM T83391 CWJ3F7 53320676 IC50 = 30 nM T83391 C15ODT 53321970 IC50 = 500 nM T83391 C7L2WY 53323322 IC50 = 500 nM T83391 COA4I5 53324112 IC50 > 10000 nM T83391 C8C7LK 53324367 IC50 = 450 nM T83391 CRVU07 54580733 IC50 = 200 nM T83391 CGI6Y9 54581737 IC50 = 820 nM T83391 CBN3O8 54583700 IC50 = 290 nM T83391 CB2Q5J 54584668 IC50 = 330 nM T83391 CCBW10 54586599 IC50 = 140 nM T83391 CE7N6G 54587610 IC50 = 640 nM T83391 C3F1BX 54587611 IC50 = 350 nM T83391 CLG5A0 57390955 IC50 > 50000 nM T83391 CE08TQ 67072047 IC50 = 1000 nM T83391 C2PU4A 76311107 IC50 > 50000 nM T83391 C7D0NU 76311108 IC50 > 50000 nM T83391 CJF2M9 76311119 IC50 = 9700 nM T83391 CQB2Y7 76311120 IC50 > 50000 nM T83391 C81MLZ 76311121 IC50 = 25600 nM T83391 CB76GD 76311122 IC50 = 3400 nM T83391 C9BJ0G 76314728 IC50 = 3700 nM T83391 CCY3D1 76314729 IC50 = 4060 nM T83391 C3PCL7 76314730 IC50 = 10300 nM T83391 CK3V9I 76314731 IC50 > 50000 nM T83391 CDH61M 76318290 IC50 > 50000 nM T83391 CN02MK 76318291 IC50 > 50000 nM T83391 C2Z6WM 76318292 IC50 > 50000 nM T83391 CP5MU2 76318293 IC50 > 50000 nM T83391 C0NVT2 76318305 IC50 > 50000 nM T83391 CF41ZJ 76321984 IC50 = 4300 nM T83391 C32LGH 76321992 IC50 = 18500 nM T83391 C4KTC9 76321993 IC50 = 35600 nM T83391 CS1Y7O 76321994 IC50 = 4500 nM T83391 CAU1L9 76321995 IC50 > 50000 nM T83391 CU8Q5Z 76325609 IC50 = 33900 nM T83391 CO4PN5 76325621 IC50 > 50000 nM T83391 CP08VY 76325622 IC50 = 7400 nM T83391 CYL3P2 76329176 IC50 > 50000 nM T83391 CNSU74 76329192 IC50 = 5400 nM T83391 CVZ90B 76329193 IC50 > 50000 nM T83391 CSFE49 76329194 IC50 = 29100 nM T83391 CAN9H0 76329195 IC50 > 50000 nM T83391 CRIP82 76329196 IC50 > 50000 nM T83391 C3UYR6 76332837 IC50 = 990 nM T83391 C30AIW 76332838 IC50 > 50000 nM T83391 CN82TO 76332850 IC50 = 7700 nM T83391 CYW5A8 76332851 IC50 = 12200 nM T83391 C74FTH 76336458 IC50 > 50000 nM T83391 CPJ27E 76336459 IC50 > 50000 nM T83391 CN0FD3 76336460 IC50 = 25900 nM T83391 C7E2ID 76336461 IC50 > 50000 nM T83391 C09FVZ 76336466 IC50 > 50000 nM T83391 C6LN4M 85770095 IC50 = 900 nM T83391 CW3G0N 85770099 IC50 = 140 nM T83391 CS1E9R 85770100 IC50 = 1900 nM T83391 C9N2IX 85770102 IC50 = 170 nM T83391 C4SC9T 85770121 IC50 = 260 nM T83391 C6YVE2 85770147 IC50 = 210 nM T83391 CJBY35 85770164 IC50 = 4000 nM T83391 CMR21T 85770169 IC50 = 70 nM T83391 CP3S5U 85770299 IC50 = 10000 nM T83391 CVK1U0 90665554 IC50 = 30 nM T83391 C8XKL9 90665555 IC50 = 1000 nM T83391 CK3A4L 90665556 IC50 = 855 nM T83391 CDL8Y9 90665557 IC50 = 6000 nM T83391 C5NDG7 90665558 IC50 = 320 nM T83391 CAER75 90665559 IC50 = 160 nM T83391 CU0MI4 90665560 IC50 = 110 nM T83391 CELR14 90665561 IC50 = 120 nM T83391 C8NG3T 90665562 IC50 = 67 nM T83391 CA5VY9 90665563 IC50 = 38 nM T83391 CX3V7A 90665707 IC50 = 40 nM T83391 CN0YD9 90665708 IC50 = 85 nM T83391 C0KX2M 90665709 IC50 = 10000 nM T83391 C5NX9R 90665710 IC50 = 2100 nM T83391 CS9I6D 90665711 IC50 = 2200 nM T83391 CX72OY 90665712 IC50 = 4300 nM T83391 C8B1SG 90665713 IC50 = 950 nM T83391 C9GCS7 90665714 IC50 = 10000 nM T83391 CI8YQ7 90665715 IC50 = 6700 nM T83391 CLH5Z3 90665716 IC50 = 10000 nM T83391 CS35GX 90665717 IC50 = 10000 nM T83391 CNR20V 118725794 IC50 = 5170 nM T83391 C0SH8Y 118725795 IC50 = 880 nM T83391 C5A9LI 118725796 IC50 = 2070 nM T83391 C94HVL 118725797 IC50 = 1290 nM T83391 C2E7VI 118725798 IC50 > 50000 nM T83391 CE3Q1N 118725799 IC50 > 50000 nM T83391 CP8QC7 118725800 IC50 > 50000 nM T83391 CIR31Y 118725801 IC50 > 50000 nM T83391 CFR9T5 118725802 IC50 = 1400 nM T83391 CEK17V 118725803 IC50 = 2400 nM T83391 CK6N2A 118725804 IC50 = 5270 nM T83391 COTI97 118725805 IC50 = 2400 nM T83391 CXM8W7 118725806 IC50 = 5220 nM T83391 C6E1TO 118725807 IC50 = 1800 nM T83391 CT8Y6B 118725808 IC50 = 1100 nM T83391 CKT1Y0 118725809 IC50 = 2000 nM T83391 CLQO31 118725810 IC50 = 2760 nM T83391 CD1X2P 118725811 IC50 = 690 nM T83391 CCR8Z9 118725812 IC50 = 690 nM T83391 C32NOW 118725813 IC50 = 1310 nM T83391 CE08CX 118725814 IC50 = 1700 nM T83391 CD92AU 118725815 IC50 = 6430 nM T83391 CQ85AX 118725816 IC50 = 450 nM T83391 CZS43L 118725817 IC50 = 100 nM T83391 CD5B6C 118725818 IC50 = 1600 nM T83391 CS0J7E 155510451 IC50 = 790 nM T83391 C2FQU8 155510458 IC50 = 1800 nM T83391 CFH0E3 155516658 IC50 = 3100 nM T83391 C6CB4E 155523516 IC50 = 840 nM T83391 C9B2FM 155530229 IC50 = 830 nM T83391 COQA96 155533655 IC50 = 640 nM T83391 C48EZG 155537837 IC50 = 2700 nM T83391 CHXY47 155539423 IC50 = 1600 nM T83391 CL87MV 155549717 IC50 = 7000 nM T83391 C75UCJ 155553477 IC50 = 5400 nM T83391 CGO9U5 155561258 IC50 = 8200 nM T83391 C54SAH 155563959 IC50 = 1600 nM T83391 C83DZW 155564495 IC50 = 2900 nM T83391 D00XCL 24856357 IC50 = 1600 nM T83391 D01RPM 11645581 IC50 = 58000 nM T83391 D07UYV 2857 IC50 = 1700 nM T83391 D0G9KD 5328245 IC50 = 7500 nM T83391 D0H6WG 44587908 IC50 = 10589 nM T83391 D0X6YR 44410037 IC50 = 7700 nM T83391 D0ZH1U 2051 IC50 = 1300 nM T81358 D03ISJ 135564632 IC50 = 3.4 nM T81358 D0LL4Y 135564531 IC50 = 17 nM T81358 D0P1CV 46191454 IC50 > 10000 nM T81358 D0Q9UX 16718576 IC50 > 10000 nM T81358 D03BNU 59604787 IC50 > 3500 nM T81358 CO0Q6N 621901 IC50 = 30 nM T81358 CIW3E8 939111 IC50 = 1.4 nM T81358 C7HBP6 10429593 IC50 > 10000 nM T81358 CNO5G6 11149390 IC50 = 20 nM T81358 CNLK30 11185393 IC50 = 178 nM T81358 COC65V 11207259 IC50 = 6 nM T81358 C2SXA0 11210036 IC50 = 19 nM T81358 CU90KX 11266364 IC50 = 64 nM T81358 C3I7WJ 11267154 IC50 = 220 nM T81358 CXS29A 11267850 IC50 = 7 nM T81358 C3F6UB 11300082 IC50 = 7 nM T81358 C4OSD3 11311779 IC50 = 12 nM T81358 CX6A1B 11347930 IC50 = 655 nM T81358 C3S2FX 11357740 IC50 = 13 nM T81358 CC8D1J 11380404 IC50 = 2 nM T81358 CUHW37 11402137 IC50 = 2 nM T81358 C6T0LA 11404817 IC50 = 262 nM T81358 C57WFQ 11425051 IC50 = 26 nM T81358 CE5R6Q 11425728 IC50 = 259 nM T81358 CU4QZ9 11483024 IC50 = 8 nM T81358 CARE96 11483025 IC50 = 636 nM T81358 CKPF03 11500189 IC50 = 5 nM T81358 CRC72L 11514482 IC50 = 45 nM T81358 CN24FK 11557879 IC50 = 14 nM T81358 CP3C1Q 11630374 IC50 = 9 nM T81358 C85TSO 11630500 IC50 = 3 nM T81358 CIJL20 11658652 IC50 = 10 nM T81358 CZX27J 11716463 IC50 = 6 nM T81358 C9JT4S 11847343 IC50 = 1970 nM T81358 C9VC3B 16202187 IC50 = 44 nM T81358 CNUL28 16661285 IC50 = 10 nM T81358 CSON67 16720432 IC50 = 147 nM T81358 CI6P4Q 16747641 IC50 = 9 nM T81358 C6H0EI 19754146 IC50 = 4700 nM T81358 C40NAR 22038513 IC50 > 5000 nM T81358 CVJX92 23582514 IC50 = 12 nM T81358 C1BLP4 23582519 IC50 = 11 nM T81358 C4LTN6 23582592 IC50 = 3 nM T81358 C85COH 23582657 IC50 = 4 nM T81358 CG57WQ 23585099 IC50 = 3300 nM T81358 CD2H9U 23585102 IC50 = 67 nM T81358 CQ9PL3 23585103 IC50 = 160 nM T81358 C06TNP 23585146 IC50 = 88 nM T81358 C8AE5G 23585147 IC50 = 5 nM T81358 CN3L2M 23585148 IC50 = 8 nM T81358 C7AB2V 23585149 IC50 = 47 nM T81358 C62PWM 23585151 IC50 = 12 nM T81358 CZ3I8N 23585152 IC50 = 23 nM T81358 C6JP1R 23585193 IC50 = 13 nM T81358 C0V5TH 23585194 IC50 = 138 nM T81358 C40VHJ 23585198 IC50 = 3 nM T81358 CR0T8H 23585200 IC50 = 42 nM T81358 CO15NZ 23585244 IC50 = 4 nM T81358 C7XZ4Q 23585245 IC50 = 404 nM T81358 C6H2XJ 23585246 IC50 > 5000 nM T81358 CPYB16 23585248 IC50 = 120 nM T81358 C6Q2NK 23585292 IC50 > 5000 nM T81358 C19-FEB 23585295 IC50 = 14 nM T81358 CI2W5O 24759475 IC50 = 150 nM T81358 CV8G9X 24759479 IC50 = 100 nM T81358 CYPF84 24759580 IC50 = 110 nM T81358 CH0W9B 24759581 IC50 = 10 nM T81358 C8W1HA 24759582 IC50 = 5 nM T81358 C16KAD 24759583 IC50 = 6 nM T81358 CD98UV 24759684 IC50 = 350 nM T81358 C0D5ZS 24759685 IC50 = 40 nM T81358 CXJ05P 24771196 IC50 = 27 nM T81358 CB3I7Y 24776677 IC50 > 5000 nM T81358 COWV67 24776678 IC50 = 28 nM T81358 CTN9U5 24776679 IC50 = 4 nM T81358 CSK01C 24776788 IC50 > 5000 nM T81358 C8UWB0 24776789 IC50 = 863 nM T81358 CB3M8A 24776790 IC50 = 1397 nM T81358 C16FNW 24778303 IC50 = 201 nM T81358 CBW78G 24778304 IC50 = 158 nM T81358 CG67XV 24778425 IC50 = 323 nM T81358 C3NF0I 24809690 IC50 = 8 nM T81358 CYX9Q0 24809691 IC50 = 23 nM T81358 CVUK80 24809692 IC50 = 14 nM T81358 CK9W8G 24809694 IC50 = 162 nM T81358 CF1I8D 24809724 IC50 = 60 nM T81358 CBV5A8 24809725 IC50 = 58 nM T81358 CGFV40 24809726 IC50 = 23 nM T81358 C5CJS7 24809727 IC50 = 39 nM T81358 CINX87 24809728 IC50 = 44 nM T81358 C9QMJ6 24809762 IC50 = 8 nM T81358 CUY8O2 24809901 IC50 = 39 nM T81358 C3HM0U 24809902 IC50 = 22 nM T81358 C0C3BN 24809931 IC50 = 5 nM T81358 CBHO82 24809932 IC50 = 2 nM T81358 CDE86V 24809933 IC50 = 52 nM T81358 CW3H2T 24809936 IC50 = 410 nM T81358 CBX41V 24809937 IC50 = 18 nM T81358 C6ZN2T 24809963 IC50 = 38 nM T81358 C4EG8R 24993189 IC50 > 10000 nM T81358 CQCU59 25108998 IC50 = 730 nM T81358 CHS70A 25109769 IC50 = 1200 nM T81358 C2CXU0 25164676 Ki = 0.5012 nM T81358 CMS6Y3 25190881 IC50 = 13 nM T81358 C41IBW 25190882 IC50 = 6 nM T81358 C37VBJ 25190883 IC50 = 5 nM T81358 C9RZ1G 25190884 IC50 = 3 nM T81358 CCVD80 25190885 IC50 = 32 nM T81358 C7ZE2X 25190887 IC50 = 11 nM T81358 C28XGU 25190888 IC50 = 10 nM T81358 C9W3DX 25190889 IC50 = 3 nM T81358 C43GEU 25190890 IC50 = 2 nM T81358 C3PX1H 25190891 IC50 = 20 nM T81358 CN8VA1 25190892 IC50 = 5 nM T81358 CIN53D 25190893 IC50 = 2 nM T81358 CZR56P 25190894 IC50 = 7 nM T81358 C0DW7B 25190895 IC50 = 24 nM T81358 CL1Q0M 25190896 IC50 = 5 nM T81358 C0AZH7 25190897 IC50 > 5000 nM T81358 CRQ5C9 25190898 IC50 = 210 nM T81358 CXT5J1 25190899 IC50 = 290 nM T81358 CL2BZ7 25194016 IC50 = 52 nM T81358 CNG96H 25210579 IC50 > 10000 nM T81358 CE93VP 44580795 IC50 = 2 nM T81358 C2G9AH 44586850 IC50 = 7300 nM T81358 C0H1JN 44586907 IC50 > 13000 nM T81358 C5BF9S 44586908 IC50 = 1000 nM T81358 CROT59 46871772 IC50 = 210 nM T81358 C9A3RQ 49787821 IC50 = 456 nM T81358 CBNA35 49787824 IC50 = 530 nM T81358 CM74QD 49787826 IC50 = 793 nM T81358 C84OLM 49787828 IC50 = 40 nM T81358 CCR9Y5 49787901 IC50 = 640 nM T81358 COY50P 49787902 IC50 = 1146 nM T81358 CV68UF 49788212 IC50 = 197 nM T81358 C8G9CU 49788553 IC50 = 516 nM T81358 C82FBN 49788554 IC50 = 482 nM T81358 CM3F4K 49788555 IC50 = 463 nM T81358 CGFZ07 49788557 IC50 = 4800 nM T81358 CLG81J 49788559 IC50 = 859 nM T81358 C5K7CJ 49788628 IC50 = 293 nM T81358 CJBG97 49788629 IC50 > 10000 nM T81358 C9LRF4 49788630 IC50 = 200 nM T81358 CHU8Q9 49788635 IC50 = 56 nM T81358 C4ZA5G 49788636 IC50 = 73 nM T81358 CSO3H2 49788704 IC50 = 53 nM T81358 CM42SG 49788705 IC50 = 412 nM T81358 CK7YT9 49788706 IC50 = 82 nM T81358 C8K1DI 49788707 IC50 = 90 nM T81358 CR0X2P 49788708 IC50 = 68 nM T81358 CR95VU 49788710 IC50 = 1300 nM T81358 CNF0T7 49788712 IC50 > 10000 nM T81358 C0U5TK 49788785 IC50 > 10000 nM T81358 CN7A5J 49788786 IC50 > 10000 nM T81358 CT96RW 49788790 IC50 = 136 nM T81358 CU1AI0 49788792 IC50 = 126 nM T81358 CZL5T8 49788860 IC50 = 117 nM T81358 CQ2P0O 49788861 IC50 = 131 nM T81358 CE69CN 49788862 IC50 = 216 nM T81358 CH47BX 49788864 IC50 = 325 nM T81358 CME3W0 49788865 IC50 = 269 nM T81358 CHM2P0 49788931 IC50 = 658 nM T81358 CE20FT 49788932 IC50 = 114 nM T81358 CI5XG9 49788933 IC50 = 68 nM T81358 C60BMA 49788936 IC50 = 280 nM T81358 C9ESQ4 49788937 IC50 = 140 nM T81358 CB19HD 49788938 IC50 = 36 nM T81358 CKYX24 49830272 Ki = 0.1585 nM T81358 CVM6X8 49830280 Ki = 0.3162 nM T81358 C3X6DN 49830474 Ki = 0.7943 nM T81358 CO98FI 49843482 Ki = 0.9 nM T81358 CE1ZK6 54759168 IC50 > 10000 nM T81358 CAK91L 56955954 IC50 > 3600 nM T81358 CYW80O 57392258 Ki = 0.28 nM T81358 CSZA16 60155724 IC50 > 3600 nM T81358 CQ8PY7 66743332 IC50 > 1000 nM T81358 C09MPF 66743431 IC50 = 290 nM T81358 CQ8PM7 66743626 IC50 > 1000 nM T81358 CSI5P9 66887486 Ki = 1.4 nM T81358 C98ARV 66888114 Ki = 5.5 nM T81358 C4SYB1 66888175 Ki = 13 nM T81358 CI9NP4 66888458 Ki = 27 nM T81358 C2AO3Q 66888604 Ki = 7.7 nM T81358 CCQP38 66888945 Ki = 67 nM T81358 CWS06D 66888952 Ki = 8.7 nM T81358 CY4S7F 66900677 Ki = 15 nM T81358 CNH3R2 68388345 IC50 = 156 nM T81358 C5L0SQ 68388404 IC50 = 66 nM T81358 C17PFG 71527115 Ki = 3.2 nM T81358 C85KAF 71527116 Ki = 1.7 nM T81358 C0PY2I 71527117 Ki = 3.4 nM T81358 CAP8U6 71553522 IC50 = 9 nM T81358 C53UOG 71560541 IC50 = 350 nM T81358 CQ25SH 71580632 IC50 = 75 nM T81358 C83CTB 71580633 IC50 = 25 nM T81358 C5D4KV 71580634 IC50 = 10400 nM T81358 C91YEO 71580635 IC50 = 9000 nM T81358 CYW8T4 71580636 IC50 = 2700 nM T81358 C6BE2H 71580637 IC50 = 8800 nM T81358 CLR9Q7 71580638 IC50 = 1500 nM T81358 CH7C2T 71580737 IC50 = 82 nM T81358 CEO1Y5 71580738 IC50 = 1100 nM T81358 C92OVF 71580739 IC50 = 3300 nM T81358 CS5DB9 71580740 IC50 = 760 nM T81358 CI7M6B 71580741 IC50 = 8500 nM T81358 CF14UA 71580742 IC50 = 26700 nM T81358 C5WGV3 71580743 IC50 = 930 nM T81358 C5JYS4 71580744 IC50 = 980 nM T81358 CU9LY4 71580745 IC50 = 12600 nM T81358 C4O5VB 71580746 IC50 = 1240 nM T81358 CYZM69 71580828 IC50 = 360 nM T81358 CN8BT6 71580829 IC50 = 5300 nM T81358 CMS1Y7 71580830 IC50 = 104 nM T81358 CV3K1J 71580831 IC50 = 160 nM T81358 C9DJ3E 71580832 IC50 = 250 nM T81358 CG32TU 71580833 IC50 = 580 nM T81358 CKZ6E1 71580834 IC50 = 120 nM T81358 CME5Z4 71580835 IC50 = 160 nM T81358 CMAC67 71580913 IC50 = 11 nM T81358 CH54UK 71580914 IC50 = 160 nM T81358 C6D3HR 71580915 IC50 = 330 nM T81358 C95XJE 71580916 IC50 = 7 nM T81358 C8R9OC 71580917 IC50 = 30 nM T81358 CGA36U 72547516 IC50 = 3200 nM T81358 C4MG8E 72547517 IC50 > 50000 nM T81358 CPA74W 72547518 IC50 > 50000 nM T81358 C4T0JS 72547519 IC50 > 50000 nM T81358 CE1VB4 72696779 IC50 = 284 nM T81358 CP26UC 76313690 IC50 = 710 nM T81358 C0Y8ZK 91933875 IC50 > 1000 nM T81358 C46KZG 131704449 IC50 = 60 nM T81358 CCPZ70 131704452 IC50 > 10000 nM T81358 CSNE45 135461314 IC50 = 2000 nM T81358 CJ36IY 135550168 IC50 = 50 nM T81358 CH2YR7 135566648 IC50 = 7.7 nM T81358 CPK76N 135712476 IC50 = 66 nM T81358 CZYX89 135712480 IC50 = 105 nM T81358 CW9BM8 135712506 IC50 = 21 nM T81358 CH90LE 135712510 IC50 = 20 nM T81358 CUE95G 135712512 IC50 = 37 nM T81358 C1K0SP 135712514 IC50 = 24 nM T81358 C85XGY 135712516 IC50 = 15 nM T81358 C10AGM 135712518 IC50 = 33 nM T81358 CF1B9J 135712520 IC50 = 18 nM T81358 CN3PL7 135712530 IC50 = 21 nM T81358 C2F3BZ 135712532 IC50 = 35 nM T81358 C6E3IN 135712534 IC50 = 247 nM T81358 CB9F1W 135712536 IC50 = 64 nM T81358 COB0T6 135712544 IC50 = 45 nM T81358 CCYM49 135712590 IC50 = 13 nM T81358 C2EW4H 135712610 IC50 = 30 nM T81358 C0LS6V 135712611 IC50 = 47 nM T81358 C0LC5W 135712618 IC50 = 60 nM T81358 C7RV8W 135712632 IC50 = 47 nM T81358 CR4AI7 135712638 IC50 = 25 nM T81358 C7MKT4 135862898 IC50 = 580 nM T81358 C5J2QN 135862901 IC50 = 7100 nM T81358 C9JBD1 135867931 IC50 = 13 nM T81358 CEX54P 135867940 IC50 = 207 nM T81358 C4XA7O 135867941 IC50 = 625 nM T81358 C7JP3T 135867977 IC50 = 9.1 nM T81358 CST7X3 135870706 IC50 = 9 nM T81358 CP2HA1 135914540 IC50 = 10 nM T81358 C1H6MX 135914549 IC50 = 4 nM T81358 C64PNW 135914550 IC50 = 26 nM T81358 CYTA89 135930672 IC50 = 3.7 nM T81358 CDI6B7 135950267 IC50 > 10000 nM T81358 CZ3RF0 135950271 IC50 = 21 nM T81358 C3N7GO 135950278 IC50 = 13 nM T81358 C6VF4N 135986108 IC50 > 10000 nM T81358 CYT69U 135986109 IC50 = 130 nM T81358 CHA4N2 136013680 IC50 > 10 nM T81358 CQY0C7 136189673 IC50 = 7.7 nM T81358 CC52HL 136189674 IC50 = 5.5 nM T81358 C8JW7N 136189743 IC50 = 2200 nM T81358 CQGO78 136189786 IC50 = 11 nM T81358 C5N2QZ 136189800 IC50 = 6.2 nM T81358 CC40LU 136189802 IC50 = 15 nM T81358 CU04TN 136189823 IC50 > 3000000 nM T81358 C4BAC9 136189831 IC50 = 14000 nM T81358 C7BU1C 136189837 IC50 > 3000000 nM T81358 CO8B4N 136189863 IC50 = 11 nM T81358 C79OQZ 136189864 IC50 = 104000 nM T81358 CJ57SF 136189870 IC50 = 3.9 nM T81358 CX3H0P 136189910 IC50 = 1350000 nM T81358 C91DKS 136189955 IC50 = 9000 nM T81358 CB6EY8 136189986 IC50 = 167 nM T81358 CCWV39 136189998 IC50 = 7.9 nM T81358 C9SP0D 136190004 IC50 = 6.1 nM T81358 CZ1DH2 136190005 IC50 = 4592 nM T81358 CYR45B 136190013 IC50 = 4.8 nM T81358 CJ5LB9 136190029 IC50 = 3.7 nM T81358 CU0MZ9 136190070 IC50 = 7.3 nM T81358 C1YUD0 136219394 IC50 > 10 nM T81358 C13FTU 136240093 IC50 = 130 nM T81358 C9XG6P 136240262 IC50 = 13000 nM T81358 C19QPI 136240263 IC50 = 140 nM T81358 CQCW57 136240264 IC50 = 51 nM T81358 C7YR3A 136240265 IC50 = 32 nM T81358 COX87S 136244262 IC50 > 3000000 nM T81358 C3RY9E 136245066 IC50 = 6200 nM T81358 C09EIK 136245067 IC50 = 150 nM T81358 CIE3Q9 136245068 IC50 = 250 nM T81358 C3F9VT 136245295 IC50 = 690 nM T81358 CGVP23 136245296 IC50 = 2600 nM T81358 CPU1F9 136245297 IC50 = 20 nM T81358 CT5IE9 136247011 IC50 = 12000 nM T81358 CE6O2S 136247012 IC50 = 370 nM T81358 CBH13D 136247014 IC50 = 71 nM T81358 CBTA26 136247015 IC50 = 60 nM T81358 C1OH4L 136247058 IC50 = 780 nM T81358 CW8HO7 136247059 IC50 = 1600 nM T81358 CJM9G0 136254209 IC50 = 1000 nM T81358 CIU8W3 136254389 IC50 > 10 nM T81358 C5YBA1 136333907 IC50 = 250 nM T81358 CJC89A 136333957 IC50 = 36 nM T81358 C1RSV0 136443837 IC50 = 67 nM T81358 C03JDR 136603225 IC50 = 41 nM T81358 CG60AI 136603274 IC50 = 350 nM T81358 CGB8T4 137645179 IC50 = 40 nM T81358 CNH56X 137648287 IC50 > 1000 nM T81358 C5KB6I 137661818 IC50 > 1000 nM T81358 CQ82UE 137662204 IC50 = 10000 nM T81358 CKEP96 155512073 IC50 = 130 nM T81358 CQ2C0D 135712546 IC50 = 18 nM T81358 CU90WN 135712554 IC50 = 39 nM T81358 C6G2JR 135712556 IC50 = 86 nM T81358 CO9B7S 135712560 IC50 = 55 nM T81358 C7QY4L 135712562 IC50 = 50 nM T81358 CL03DP 135712564 IC50 = 162 nM T81358 C6NTO1 135712588 IC50 = 207 nM T81358 C16WXV 135950266 IC50 = 128 nM T81358 C5DF6L 135950268 IC50 = 116 nM T81358 CFRA48 135950274 IC50 > 10000 nM T81358 C9RAM5 135950279 IC50 = 238 nM T81358 CE9D5W 135950285 IC50 = 127 nM T81358 D03DZO 11715767 IC50 = 10 nM T81358 D08HFG 24809764 IC50 = 22 nM T81358 D09HVH 135566652 IC50 > 10 nM T81358 D0T8NU 16757525 IC50 = 2 nM T53468 D02KKA 24856436 IC50 = 2310 nM T53468 CN8WB9 44189332 IC50 = 401 nM T53468 CV63UL 67240318 IC50 > 10000 nM T53468 CXC69T 137321158 IC50 = 97 nM T53468 C2MD1Q 155513187 IC50 > 10000 nM T53468 D0E7VO 59627005 IC50 = 99.8 nM T98091 D05HSW 3218 Ki = 23.6 nM T98091 CUOK35 1563 Ki = 318 nM T98091 CGX91W 3071 EC50 = 252 nM T98091 C1S4PG 16064 EC50 = 432 nM T98091 CWY93I 37289 EC50 > 100000 nM T98091 CV13DQ 73015 Ki > 10000 nM T98091 CXH9K8 169433 EC50 > 100000 nM T98091 C6PKO7 182326 EC50 >= 10000 nM T98091 CU79RS 254323 EC50 > 10000 nM T98091 CUR6F9 308653 Ki = 10.8 nM T98091 CIK92G 308775 Ki = 3.12 nM T98091 C7BV2W 309844 Ki = 0.58 nM T98091 CS5R8E 309859 Ki = 2.1 nM T98091 C0BP6D 309900 Ki = 91 nM T98091 CPA6N4 345521 EC50 > 10000 nM T98091 CN5L4P 660705 EC50 = 2480 nM T98091 CE84YW 713598 EC50 > 10000 nM T98091 CDMV21 1912564 Ki = 0.219 nM T98091 C0YE6L 2778732 EC50 = 2970 nM T98091 C7UY3F 2940609 EC50 > 10000 nM T98091 C0K1ZQ 5302583 EC50 > 10000 nM T98091 COT13S 5312743 EC50 > 100000 nM T98091 C7ASQ0 5312744 EC50 > 100000 nM T98091 CMC0W2 6452189 EC50 > 10000 nM T98091 C3MH9Q 6516560 EC50 > 10000 nM T98091 CO12XI 9856798 EC50 >= 10000 nM T98091 C6E3TY 9878666 IC50 = 14000 nM T98091 C5O0XE 9882204 EC50 = 80 nM T98091 C25KUF 9901435 EC50 = 250 nM T98091 CTY3X1 9944370 EC50 = 103 nM T98091 CNZ5W7 10176767 EC50 > 100000 nM T98091 C5V3CB 10201214 EC50 = 59.1 nM T98091 CZ2TJ7 10266133 EC50 = 6070 nM T98091 CS62HG 10903823 EC50 > 10000 nM T98091 CEW03D 11150029 EC50 = 2970 nM T98091 C2FQ9U 11162554 EC50 > 10000 nM T98091 CK9F7Z 11359757 EC50 > 10000 nM T98091 CFGD08 11371604 EC50 > 10000 nM T98091 CWR98I 11507535 EC50 = 7290 nM T98091 CE1XJ4 12037446 EC50 = 2270 nM T98091 C6TP3C 12178423 EC50 > 10000 nM T98091 C4E2GZ 12380289 EC50 = 553 nM T98091 CU89DK 12782103 Ki = 37 nM T98091 CJOA47 13413723 EC50 = 264 nM T98091 CBJ23P 14454530 EC50 > 100000 nM T98091 CRJC57 15549641 Ki = 3470 nM T98091 CXKZ29 15949125 EC50 > 10000 nM T98091 C6S7BZ 16749196 EC50 > 10000 nM T98091 CUO75A 21204487 Ki = 469 nM T98091 C4R2KU 23042624 EC50 = 454 nM T98091 C32HZQ 23439046 EC50 > 10000 nM T98091 CIA3X8 23699039 EC50 = 38018.94 nM T98091 CY42RJ 24205051 EC50 >= 10000 nM T98091 C6WUZ8 44244396 EC50 >= 10000 nM T98091 CO8F0D 44349289 Ki = 0.726 nM T98091 CJ4N9E 44349321 Ki = 2.98 nM T98091 C8YFD1 44551836 EC50 > 10000 nM T98091 C8BKL6 53996334 EC50 > 10000 nM T98091 CBG21Q 54678947 EC50 = 1.26 nM T98091 CM42GU 56933638 EC50 > 10000 nM T98091 C4ZU6W 69454902 EC50 > 10000 nM T98091 CPDU72 70233802 EC50 = 3669 nM T98091 CJ0P4L 70521246 Ki = 1210 nM T98091 CVD73P 71442476 EC50 > 10000 nM T98091 CH2LO1 72711216 EC50 = 302 nM T98091 CBM6A2 86293760 Ki = 497 nM T98091 C2KBC9 101999730 EC50 >= 10000 nM T98091 CYZJ96 102219032 EC50 = 987 nM T98091 C7PCS5 102219035 EC50 = 5340 nM T98091 CYH40T 102338889 EC50 > 100000 nM T98091 CXHS35 102583156 EC50 = 495 nM T98091 C42TWQ 110698276 Ki = 1590 nM T98091 C49ART 110698284 Ki = 1560 nM T98091 C1W6TS 114333799 EC50 > 100000 nM T98091 CY2N8Q 121205397 Ki = 49.4 nM T98091 CX1ZQ0 127043349 EC50 = 641 nM T98091 C8Q7WT 127043463 EC50 = 3860 nM T98091 CGEK43 127043533 EC50 = 231 nM T98091 CT8EI5 127043534 EC50 = 1160 nM T98091 C5N9OI 127043659 EC50 > 100000 nM T98091 CG4W0T 127044004 EC50 = 1080 nM T98091 C53SFD 127044143 EC50 = 12.7 nM T98091 CI4UO6 127044147 EC50 > 100000 nM T98091 CBRI24 127044148 EC50 = 2105 nM T98091 CC5Y7M 127044149 EC50 = 11.4 nM T98091 C9JRX8 127044150 EC50 = 299 nM T98091 C9EBS6 127044151 EC50 = 88.1 nM T98091 CN2MJ1 127044155 EC50 = 1.34 nM T98091 CR2XE6 127044299 EC50 = 6.14 nM T98091 CBTJ96 127044300 EC50 = 811 nM T98091 C0J2UY 127044463 EC50 = 271 nM T98091 C0IFB9 127044607 EC50 = 48.7 nM T98091 CH1LK6 127044950 EC50 = 8850 nM T98091 CG0FY6 127045103 Ki = 0.324 nM T98091 C3T1DR 127045328 EC50 > 100000 nM T98091 CP3D5Y 127045422 EC50 = 0.189 nM T98091 CR57ZO 127045477 EC50 = 25700 nM T98091 CRE1X8 127045478 EC50 = 11300 nM T98091 CXYI69 127045479 EC50 = 21600 nM T98091 C2HZK7 127045480 EC50 = 653 nM T98091 C8QZP5 127045481 EC50 = 938 nM T98091 CMI92X 127045482 EC50 = 43400 nM T98091 CP26VZ 127045483 EC50 > 100000 nM T98091 CCJ94H 127045484 EC50 > 100000 nM T98091 CX2D7R 127045635 Ki = 0.7 nM T98091 CKSY93 133081959 Ki = 0.317 nM T98091 CB1GH3 135412234 Ki = 3630 nM T98091 C70QAJ 135458798 EC50 > 100000 nM T98091 C2JS0V 136342296 Ki > 10000 nM T98091 COT26K 136342308 Ki = 145 nM T98091 CM92JS 136986925 EC50 > 100000 nM T98091 CJ7NG6 137205240 EC50 > 100000 nM T98091 CEL98H 137205241 EC50 > 100000 nM T98091 CPK4I5 137205242 EC50 > 100000 nM T98091 CUYP35 137631992 EC50 > 10000 nM T98091 C6UNP5 137632827 EC50 = 175 nM T98091 C01JUA 137634047 IC50 = 10 nM T98091 CIP7O3 137635702 EC50 = 61.8 nM T98091 C6F7OM 137636801 IC50 = 10 nM T98091 CU9PN5 137639966 EC50 > 10000 nM T98091 CZN62O 137641006 EC50 > 10000 nM T98091 CL7X4V 137641589 EC50 > 10000 nM T98091 CT24MX 137642690 EC50 >= 10000 nM T98091 CI7PS8 137643534 IC50 = 10 nM T98091 C0P8SL 137643701 EC50 = 41.3 nM T98091 CA1GQ8 137644031 EC50 > 10000 nM T98091 C5XYS9 137647203 IC50 = 10 nM T98091 CO86MV 137648721 IC50 = 10 nM T98091 C2UPH8 137648861 EC50 > 10000 nM T98091 CN9V7H 137649231 EC50 = 264 nM T98091 C79TSC 137649817 EC50 = 52.4 nM T98091 CDS94V 137652440 IC50 = 10 nM T98091 CK9JZ7 137653608 EC50 > 10000 nM T98091 CZ14EN 137654126 EC50 = 83.6 nM T98091 C5UR9C 137656606 EC50 = 10000 nM T98091 CRIF83 137657052 EC50 > 10000 nM T98091 C9L2QM 137657193 IC50 = 10 nM T98091 CD9Y3C 137658184 EC50 = 129 nM T98091 C5YO8K 137658671 EC50 = 328 nM T98091 CTV96Z 137658717 EC50 > 10000 nM T98091 C7CV6H 137661584 IC50 = 10 nM T98091 C2M1JC 137661917 EC50 > 10000 nM T98091 CJR25V 140898903 Ki = 3.77 nM T98091 CVN8G7 146025740 Ki = 0.866 nM T98091 CMH04C 146025741 Ki = 1.12 nM T98091 C7VID6 146025742 Ki = 267 nM T98091 C3H1JE 146025744 Ki = 6.94 nM T98091 C9NX6Y 146025745 Ki = 3.6 nM T98091 CYGU43 146025746 Ki = 1.25 nM T98091 C6WBH0 146025747 Ki = 11.4 nM T98091 CL6W4O 146025748 Ki = 0.65 nM T98091 C24EUS 146025749 Ki = 0.582 nM T98091 CBLV13 146025751 Ki = 1.27 nM T98091 C4UA8F 146025752 Ki = 9.48 nM T98091 CW21NB 146025753 Ki = 4.75 nM T98091 CSW3U0 146025754 Ki = 3.99 nM T98091 CG7N3J 146025755 Ki = 35.6 nM T98091 C43KXG 146025756 Ki = 36 nM T98091 C3WR2E 146025758 Ki = 2.3 nM T98091 C6S0BV 146025759 Ki = 18.7 nM T98091 CU97BV 146025760 Ki = 44.4 nM T98091 CY4WO0 146025762 Ki = 58.6 nM T98091 CMW8O3 146025763 Ki = 189 nM T98091 C9W0IF 151217144 Ki >= 100000 nM T98091 CN16PE 153870611 Ki > 10000 nM T98091 C9D0WG 155513228 Ki = 2.63 nM T98091 C9XT1M 155525380 Ki = 225 nM T98091 CF95HD 155526533 Ki = 62.7 nM T98091 CH9CL1 155547589 Ki > 10000 nM T98091 C9CKI0 155549030 Ki = 3.28 nM T98091 CBD7J1 155551005 Ki = 37.4 nM T98091 C7LGZ3 155559672 Ki = 3.17 nM T98091 CZA0P9 155560912 Ki = 34.7 nM T98091 CH0YB8 155564247 Ki = 14.7 nM T98091 CBJ45X 155564383 Ki = 36.7 nM T98091 D03GHN 26612 Ki = 3310 nM T98091 D03JPL 79034 Ki > 10000 nM T98091 D06YGT 12530 EC50 = 1700 nM T98091 D08OBF 11005 Ki = 2640 nM T98091 D0A0GD 5288266 EC50 = 452 nM T98091 D0E7NO 2969 Ki = 1780 nM T98091 D0N0UC 3893 Ki = 2170 nM T98091 D0Q3QI 94180 EC50 > 100000 nM T98091 D0R1MM 10354234 Ki = 0.626 nM T98091 D0T2CG 94216 Ki = 110 nM T98091 D0T4BP 97783 EC50 = 12882.5 nM T98091 D0X0PF 8180 Ki = 108 nM T98091 D0XS4G 379 Ki = 19600 nM T67103 CDV02G 11628719 IC50 = 38800 nM T67103 CTO29I 44591126 IC50 = 2050 nM T67103 C4U9VF 44591153 IC50 = 4800 nM T67103 CER2H0 44591154 IC50 = 600 nM T67103 C7TX9N 44591155 IC50 = 4300 nM T67103 C3F9KJ 45267472 IC50 = 24 nM T67103 CUJ20F 45267473 IC50 = 208 nM T67103 CG4R1S 45267474 IC50 = 793 nM T67103 CL2BW6 45267475 IC50 = 8000 nM T67103 CT8HE3 45267529 IC50 > 50000 nM T67103 CK2Z3O 45267535 IC50 > 50000 nM T67103 C1DM6O 45267543 IC50 = 44 nM T67103 CJ5GW9 45267547 IC50 = 32 nM T67103 C1GV2I 45267553 IC50 = 260 nM T67103 CY4TR1 45267559 IC50 = 729 nM T67103 C6SV5H 45268342 IC50 = 975 nM T67103 CH5TZ4 45268343 IC50 = 78 nM T67103 CZDU14 45268344 IC50 = 260 nM T67103 CR53XL 45268415 IC50 = 120 nM T67103 C1ELU4 45268416 IC50 = 9100 nM T67103 CR0K6A 45268421 IC50 = 81 nM T67103 C1KBR4 45268435 IC50 = 25 nM T67103 C6OIB8 45268439 IC50 = 118 nM T67103 C47ZLB 45269206 IC50 = 98 nM T67103 COV61L 45269263 IC50 > 50000 nM T67103 CM6Z0K 45269265 IC50 = 8000 nM T67103 CZ3LR0 45269273 IC50 = 4600 nM T67103 CZY12B 45270076 IC50 = 700 nM T67103 CN86ZB 45270113 IC50 > 50000 nM T67103 CS90FU 45270114 IC50 > 50000 nM T67103 C3QNG5 45270128 IC50 = 8 nM T67103 C47QFS 45270947 IC50 > 50000 nM T67103 CDTM02 45270948 IC50 = 30000 nM T67103 C1C0OW 45270949 IC50 > 50000 nM T67103 C30CPF 45270951 IC50 > 50000 nM T67103 CM93NG 45270952 IC50 > 50000 nM T67103 CMX80K 45270962 IC50 = 41 nM T67103 CHM04R 45271812 IC50 = 320 nM T67103 CY06PO 45271816 IC50 = 62 nM T67103 C5GEP3 45272661 IC50 = 800 nM T67103 CA9QV5 45272669 IC50 > 50000 nM T67103 CU5WP0 45273592 IC50 > 50000 nM T67103 CUPR63 45273593 IC50 > 50000 nM T67103 CISY97 45273600 IC50 = 11 nM T67103 CL9FH7 45273601 IC50 = 63 nM T67103 CF42OQ 45273605 IC50 = 301 nM T67103 CXP53S 45273612 IC50 = 19 nM T67103 C5PZ8G 46201042 IC50 = 11000 nM T67103 C81VUL 46229417 IC50 = 5800 nM T67103 CNP0O2 46229418 IC50 = 33700 nM T67103 CPB51X 46229419 IC50 > 100000 nM T67103 CC6HP8 46229421 IC50 = 8300 nM T67103 C1CR9Y 46229422 IC50 = 4800 nM T67103 CR53AM 46229424 IC50 = 15600 nM T67103 C0PU3D 73351771 IC50 = 18800 nM T67103 CJL87N 135949396 IC50 = 5 nM T67103 CSCN42 135983770 IC50 = 14 nM T67103 CR8K5L 135983772 IC50 = 310 nM T12119 D03FLC 3878 IC50 = 17000 nM T12119 D04MSM 2554 IC50 = 22000 nM T12119 D05OFX 219078 IC50 = 182 nM T12119 D08HQK 5411 IC50 = 56 nM T12119 D0C7ET 11174599 IC50 < 30 nM T12119 D0E4DW 1775 IC50 > 100000 nM T12119 D0TV6I 131682 IC50 = 100000 nM T12119 D0X0RI 4178 IC50 = 11000 nM T12119 D0X4RN 3676 IC50 = 29000 nM T12119 D0Y5UG 2160 IC50 = 7000 nM T12119 D00BUR 216327 IC50 > 1000 nM T12119 D04JZH 11659955 IC50 = 14000 nM T12119 D0BT0Z 68109743 IC50 = 31 nM T12119 D0K9IF 71666749 IC50 > 30000 nM T12119 D0O7QA 46840946 IC50 = 8.6 nM T12119 D0P5CM 56945146 IC50 = 66 nM T12119 D0W8XT 60663 IC50 = 500 nM T12119 D0HG2S 86294663 IC50 > 30000 nM T12119 D07EQF 9816959 Ki = 360 nM T12119 C3H6AQ 21467 IC50 = 14000 nM T12119 CPN25U 998021 IC50 = 5200 nM T12119 C8ET1W 1194121 IC50 > 30000 nM T12119 CTZ4R5 2730286 IC50 = 300 nM T12119 CORX94 2804997 IC50 = 28.18 nM T12119 CIC31J 2914136 IC50 = 300 nM T12119 CY60IU 2915811 IC50 = 200 nM T12119 CM8IR4 4879545 IC50 = 31 nM T12119 C2T5QL 5297665 IC50 > 5000 nM T12119 C5FB0O 6324668 IC50 = 18.6 nM T12119 C5TF4U 9927558 Ki = 13 nM T12119 CT0RF9 9950804 IC50 = 224 nM T12119 C5NG2C 10021733 Ki = 20 nM T12119 C5WLU0 10039502 IC50 = 1810 nM T12119 CXSN58 10370036 Ki = 150 nM T12119 CBC78O 10739578 IC50 > 1000 nM T12119 CN9ID0 11152141 IC50 = 163 nM T12119 C6FX8E 11166272 Ki = 140 nM T12119 CY57GR 11187635 IC50 = 260 nM T12119 CP6UL9 11200377 Ki = 160 nM T12119 CNH49X 11231810 Ki = 0.018 nM T12119 CYE9P4 11232185 IC50 = 738 nM T12119 C4LE9X 11267659 IC50 = 2990 nM T12119 CU92SV 11268687 IC50 = 875 nM T12119 C72OZF 11278604 IC50 = 2140 nM T12119 C0RBE9 11303465 IC50 = 620 nM T12119 CWGF86 11303911 IC50 = 1370 nM T12119 CO05XK 11371458 IC50 = 2360 nM T12119 CD68AR 11380674 IC50 = 150 nM T12119 CUP3N5 11393872 IC50 = 508 nM T12119 C3CU1H 11450354 IC50 = 270 nM T12119 CPF24M 11467411 Ki = 210 nM T12119 CCX8M4 11484925 IC50 = 1800 nM T12119 CVUM08 11640384 Ki = 360 nM T12119 C0Z5JS 11740023 Ki = 15 nM T12119 CP2S0Q 11998203 IC50 = 440 nM T12119 C6ZQS1 11998204 IC50 = 3340 nM T12119 C7PW6D 11998468 IC50 = 240 nM T12119 CFSJ84 11998825 IC50 = 1180 nM T12119 CS72UI 12003986 IC50 > 5000 nM T12119 CWK36M 12003987 IC50 > 5000 nM T12119 C4CW2A 12003988 IC50 > 5000 nM T12119 C13UTR 12004047 IC50 > 5000 nM T12119 CF98QV 12004190 IC50 = 2140 nM T12119 CF9PU6 12004191 IC50 = 140 nM T12119 CSE8Y7 12004194 IC50 = 480 nM T12119 CJCK91 12004217 IC50 = 270 nM T12119 C0R4XA 12004218 IC50 = 4170 nM T12119 CFPW42 12004278 IC50 = 1580 nM T12119 C81GMS 12004337 IC50 = 30 nM T12119 CM8VJ7 12004352 IC50 = 80 nM T12119 CXFG84 12004354 IC50 = 70 nM T12119 CP2OZ0 12004357 IC50 = 130 nM T12119 CQYB52 12004359 IC50 = 90 nM T12119 CYG2T8 12004377 IC50 = 20 nM T12119 CL1TF0 12004382 IC50 > 5000 nM T12119 CBF18D 21558498 IC50 = 17 nM T12119 CVT7X4 23642326 IC50 = 192 nM T12119 CE7DV0 23661730 IC50 = 35 nM T12119 CW3C9T 24816161 IC50 = 6080 nM T12119 CW5SX8 24874622 IC50 = 34 nM T12119 CH46XE 24874708 IC50 = 57 nM T12119 C1V9IR 24874746 IC50 = 78 nM T12119 C9DB4G 24874749 IC50 = 494 nM T12119 C1F2PB 24874784 IC50 = 150 nM T12119 CH5J6Y 24874788 IC50 = 44 nM T12119 CHO5N0 24874790 IC50 = 70 nM T12119 C97JUB 24874828 IC50 = 9 nM T12119 C8QN4Z 24874829 IC50 = 98 nM T12119 C4BN5G 24874831 IC50 = 18 nM T12119 C3VT5O 24874869 IC50 = 14 nM T12119 C0MJ8C 24874870 IC50 = 23 nM T12119 CMR31Q 24874871 IC50 = 137 nM T12119 C5KXZ7 24874872 IC50 = 295 nM T12119 CZL1S9 24874912 IC50 > 1000 nM T12119 CAYI67 24874915 IC50 = 45 nM T12119 CMCQ63 24874959 IC50 = 32 nM T12119 C4QEV8 24875004 IC50 = 65 nM T12119 C2ATU3 24875008 IC50 = 131 nM T12119 CQ35UO 24875058 IC50 = 22 nM T12119 COD41K 24875059 IC50 = 177 nM T12119 C7WH4K 24875109 IC50 = 453 nM T12119 CE23KM 24875161 IC50 = 94 nM T12119 C68VHE 24875200 IC50 = 98 nM T12119 CNDC03 24875248 IC50 > 1000 nM T12119 CUW8G0 24875251 IC50 > 1000 nM T12119 CV3W1B 24875288 IC50 = 128 nM T12119 COW05T 24875291 IC50 = 203 nM T12119 C6CK5U 24883321 IC50 = 2620 nM T12119 C5WOA3 24883322 IC50 = 1880 nM T12119 CZOT73 24896609 IC50 = 30 nM T12119 CBPY64 25008621 IC50 = 80 nM T12119 CFX2G6 25031120 IC50 = 409 nM T12119 C7A3VD 25031121 IC50 = 142 nM T12119 C7HRT3 25031122 IC50 = 49 nM T12119 CCVN84 25031123 IC50 = 47 nM T12119 CH0O2Z 25031203 IC50 = 81 nM T12119 CZD5A9 25031204 IC50 = 188 nM T12119 CP94WN 25031205 IC50 = 25 nM T12119 C0C9HJ 25031207 IC50 = 102 nM T12119 CVC0S3 25031293 IC50 = 96 nM T12119 CG17JX 25031294 IC50 = 196 nM T12119 CORL19 25031387 IC50 = 75 nM T12119 C8AJ2I 25031389 IC50 = 101 nM T12119 C9APL1 25031478 IC50 = 142 nM T12119 CWZ7F0 25031566 IC50 = 131 nM T12119 CMXJ46 25031567 IC50 = 73 nM T12119 CXF0I2 25031568 IC50 = 120 nM T12119 CL64OF 25033155 Ki = 0.63 nM T12119 C9PF3W 25033156 IC50 = 149 nM T12119 C0Z2SQ 25056787 IC50 = 158.49 nM T12119 CPAZ91 25056788 IC50 = 316.23 nM T12119 C6OCA7 25064916 IC50 = 130 nM T12119 C3VG1F 25065121 IC50 > 1000 nM T12119 CZPH98 25065124 IC50 = 60 nM T12119 C9GDR3 25065329 IC50 = 180 nM T12119 CZVX23 25065529 IC50 = 4 nM T12119 CM3A1I 25065531 IC50 = 350 nM T12119 CP03LT 25113806 IC50 = 1000 nM T12119 CY5A6Q 25113809 IC50 = 1258.93 nM T12119 C95YUJ 25113810 IC50 = 1584.89 nM T12119 CK3JN1 25138309 IC50 = 9.333 nM T12119 CP72MB 25159060 IC50 = 10000 nM T12119 CXKB13 25204469 IC50 = 23.99 nM T12119 CAW05V 25204470 IC50 = 138.04 nM T12119 C38CAX 25204471 IC50 = 151.36 nM T12119 CUZ1Y2 25204472 IC50 = 22.91 nM T12119 C1GO8L 25204473 IC50 = 28.84 nM T12119 C9ZTJ3 25204533 IC50 = 72.44 nM T12119 C2O6LT 25204534 IC50 = 302 nM T12119 CBG48F 25204535 IC50 = 223.87 nM T12119 C3JN6D 25204536 IC50 = 331.13 nM T12119 CC9A3W 25204537 IC50 = 12589.25 nM T12119 C76UDL 25204600 IC50 = 162.18 nM T12119 CXOZ41 25204603 IC50 = 169.82 nM T12119 C08BDN 25204604 IC50 = 10.47 nM T12119 C4IUB3 25204605 IC50 = 38.02 nM T12119 CBH9O2 25204669 IC50 = 208.93 nM T12119 C92WAR 25204670 IC50 = 1174.9 nM T12119 CYIV75 25204736 IC50 = 4466.84 nM T12119 CZY68S 25204738 IC50 = 263.03 nM T12119 C2K5WT 44311988 IC50 > 1000 nM T12119 CMB53J 44391429 IC50 = 210 nM T12119 C7GEJ1 44391502 IC50 = 2900 nM T12119 C7Y2LN 44391503 IC50 = 3200 nM T12119 CT9A6J 44391509 IC50 > 10000 nM T12119 CW2IZ0 44391519 IC50 = 10000 nM T12119 CER59T 44391523 IC50 = 1400 nM T12119 CH4CF2 44391524 IC50 = 10000 nM T12119 CXB13I 44391527 Ki = 60 nM T12119 CGDC86 44391528 IC50 = 2900 nM T12119 C0LS6Y 44391531 IC50 = 5300 nM T12119 C6X5OS 44391532 IC50 = 2300 nM T12119 CXOC73 44391533 IC50 = 10000 nM T12119 CDM9F2 44391535 Ki = 670 nM T12119 CB7P0N 44391536 IC50 > 10000 nM T12119 C51UGS 44391538 Ki = 410 nM T12119 CL51IC 44391543 Ki = 50 nM T12119 CZ03AB 44391545 IC50 = 840 nM T12119 CUVG84 44391546 IC50 = 10000 nM T12119 CI5O0M 44391551 IC50 = 1400 nM T12119 CA6E5P 44391552 IC50 > 10000 nM T12119 C1X9EZ 44391558 IC50 = 760 nM T12119 C1XUL5 44391561 Ki = 140 nM T12119 C7JD3V 44391562 IC50 > 10000 nM T12119 CTSA82 44391568 IC50 = 860 nM T12119 C4CBU9 44391571 IC50 = 10000 nM T12119 CB56OV 44391575 Ki = 2000 nM T12119 CR1L0M 44391577 IC50 > 10000 nM T12119 C4IR6G 44391582 Ki = 110 nM T12119 CX3V8F 44391591 Ki = 280 nM T12119 CCMY53 44391601 IC50 > 10000 nM T12119 CYZ06F 44391609 IC50 = 300 nM T12119 C7ARZ6 44391618 Ki = 2500 nM T12119 CFA5R9 44391619 IC50 > 10000 nM T12119 C3N0JB 44391627 Ki = 330 nM T12119 C8WXZ6 44391630 IC50 = 5000 nM T12119 COZ87E 44391631 Ki = 130 nM T12119 C5G9HV 44391649 IC50 = 1100 nM T12119 CTF35M 44391655 Ki = 140 nM T12119 CAG4R9 44391656 Ki = 30 nM T12119 C7SVA3 44391657 Ki = 370 nM T12119 C3Z1KM 44391658 IC50 = 660 nM T12119 C2EF9D 44391663 Ki = 2100 nM T12119 C82OZY 44391664 Ki = 530 nM T12119 CSF80B 44391674 IC50 = 370 nM T12119 CDG5J3 44391682 Ki = 160 nM T12119 CIS05R 44391684 IC50 = 5000 nM T12119 CQWK68 44402348 IC50 = 730 nM T12119 CF8C6L 44402353 IC50 = 3700 nM T12119 CC4O3R 44402387 IC50 = 4000 nM T12119 CDK3R0 44402391 IC50 = 7500 nM T12119 CJC8L9 44402412 IC50 = 2200 nM T12119 CW3Y9N 44402448 IC50 = 4000 nM T12119 C08LKH 44402452 IC50 = 2900 nM T12119 CQZ4B9 44402481 IC50 = 550 nM T12119 C14WJU 44402485 IC50 = 40000 nM T12119 CQZM30 44402530 IC50 = 550 nM T12119 CQSA35 44402548 IC50 = 29000 nM T12119 CA7BT3 44402565 IC50 = 6600 nM T12119 CY2W0T 44402585 IC50 = 7400 nM T12119 CXJ0Z6 44402597 IC50 = 3800 nM T12119 CX9QB6 44402602 IC50 = 6500 nM T12119 C7ZE2M 44402626 IC50 > 30000 nM T12119 C24MBZ 44402629 IC50 = 22000 nM T12119 C26SHX 44402675 IC50 = 860 nM T12119 C7P5LA 44402679 IC50 = 19400 nM T12119 CUF6Q5 44402703 IC50 = 90000 nM T12119 CD1HW4 44402745 IC50 = 21000 nM T12119 CG61ZQ 44402807 IC50 > 30000 nM T12119 CXPD29 44402815 IC50 > 30000 nM T12119 CW4C5K 44408740 Ki = 820 nM T12119 CIW75T 44408743 Ki > 3000 nM T12119 C5IKC7 44408744 Ki = 630 nM T12119 CP3BF5 44408772 Ki = 980 nM T12119 C6V3WX 44408776 Ki = 330 nM T12119 CCZU51 44408787 Ki = 1150 nM T12119 CMPT60 44408788 Ki = 440 nM T12119 CQDU28 44408791 Ki = 440 nM T12119 CXWL81 44408928 Ki = 250 nM T12119 CX79PW 44408929 Ki = 1490 nM T12119 C7NA8C 44408932 Ki > 3000 nM T12119 C18XDS 44408933 Ki > 3000 nM T12119 CRO59N 44408937 Ki = 1110 nM T12119 CM21QY 44408938 Ki > 3000 nM T12119 C5Z3WI 44408958 Ki = 870 nM T12119 CWI4U3 44408961 Ki = 1210 nM T12119 CE89SF 44408979 Ki > 3000 nM T12119 C3KAX8 44408980 Ki = 320 nM T12119 C5U6BS 44408984 Ki = 230 nM T12119 CU3P4F 44408985 Ki > 3000 nM T12119 CQ2R0S 44442614 IC50 = 125 nM T12119 CM5N2O 44442615 IC50 > 1000 nM T12119 C34FPS 44442616 IC50 > 1000 nM T12119 CMF95A 44442617 IC50 = 375 nM T12119 CVST09 44442618 IC50 = 238 nM T12119 CA31NZ 44442619 IC50 = 87 nM T12119 C5OTW7 44442620 IC50 = 71 nM T12119 CH20PN 44442622 IC50 = 684 nM T12119 CTFR94 44442624 IC50 = 978 nM T12119 C36DVG 44442625 IC50 > 1000 nM T12119 CQL1J9 44442627 IC50 > 1000 nM T12119 C1TZD6 44442636 IC50 > 1000 nM T12119 CKE62M 44442638 IC50 > 1000 nM T12119 CJ8F0W 44442640 IC50 > 1000 nM T12119 CFIB18 44442641 IC50 > 1000 nM T12119 CR3Q7T 44442642 IC50 > 1000 nM T12119 C3B9AG 44442643 IC50 = 150 nM T12119 CKU6L5 44442644 IC50 > 1000 nM T12119 CEY38I 44442645 IC50 = 380 nM T12119 CE5V0D 44442646 IC50 = 420 nM T12119 CZJ0C7 44442647 IC50 > 1000 nM T12119 CR9T5G 44442657 IC50 > 1000 nM T12119 CY0R3M 44442661 IC50 = 145 nM T12119 CT0XB5 44442664 IC50 = 885 nM T12119 CE9DS0 44442675 IC50 = 32 nM T12119 CBQ16H 44442677 IC50 = 214 nM T12119 CSB51X 44444161 IC50 = 868 nM T12119 CC9F5I 44444174 IC50 = 175 nM T12119 C71UPR 44444177 IC50 > 1000 nM T12119 CC75RD 44444178 IC50 = 44 nM T12119 CE0KS2 44444180 IC50 = 80 nM T12119 CVT6F1 44444182 IC50 = 108 nM T12119 C2RUL0 44444186 IC50 = 169 nM T12119 C42PTL 44444190 IC50 = 146 nM T12119 CW47IU 44444192 IC50 > 1000 nM T12119 CS4KI7 44444194 IC50 = 232 nM T12119 CC2DF7 44444196 IC50 = 290 nM T12119 CCYB53 44444197 IC50 = 107 nM T12119 C5XAB1 44447254 IC50 > 10000 nM T12119 C4IGR9 44447255 IC50 > 10000 nM T12119 CQHJ42 44447256 IC50 > 10000 nM T12119 CYH4O2 44447257 IC50 = 1000 nM T12119 CL0UO5 44447258 IC50 > 1000 nM T12119 CK9UL2 44447260 IC50 = 185 nM T12119 C6IX3N 44447261 IC50 = 81 nM T12119 CHMJ82 44447262 IC50 = 123 nM T12119 C3B1OF 44447264 IC50 = 243 nM T12119 CS0ZO6 44447266 IC50 = 83 nM T12119 C8AMU9 44447267 IC50 = 255 nM T12119 C8VBD2 44447268 IC50 = 191 nM T12119 C5C3YI 44447269 IC50 = 186 nM T12119 CF90DG 44447270 IC50 = 261 nM T12119 C0WDU7 44447271 IC50 = 86 nM T12119 CHBA64 44447272 IC50 = 552 nM T12119 CUJ50E 44447273 IC50 = 129 nM T12119 C0HV4L 44447274 IC50 = 232 nM T12119 CGZ4E6 44447275 IC50 = 476 nM T12119 C4ZGH1 44447276 IC50 = 1195 nM T12119 C5MT0J 44447277 IC50 = 261 nM T12119 C7PB9V 44447278 IC50 = 181 nM T12119 CQ7AT9 44447279 IC50 = 394 nM T12119 CIY3T7 44447280 IC50 = 158 nM T12119 CP7D3U 44447281 IC50 = 132 nM T12119 CC71MI 44447282 IC50 = 148 nM T12119 CEF81H 44447283 IC50 = 221 nM T12119 CHV6W5 44447284 IC50 = 1053 nM T12119 CULB63 44447285 IC50 = 148 nM T12119 CK4Q6O 44447286 IC50 = 275 nM T12119 C0PT9W 44447287 IC50 = 171 nM T12119 C5NKU9 44447288 IC50 = 63 nM T12119 CY41VI 44447289 IC50 = 147 nM T12119 CX8GC7 44447290 IC50 = 102 nM T12119 CK6Q0S 44447291 IC50 = 158 nM T12119 CUW24D 44447292 IC50 = 744 nM T12119 CJM6O7 44447293 IC50 = 153 nM T12119 CBC5F7 44447294 IC50 = 329 nM T12119 CYB0L8 44447295 IC50 = 540 nM T12119 CHS74Q 44447296 IC50 = 182 nM T12119 CDP13B 44447605 IC50 = 219 nM T12119 C7BN0X 44447606 IC50 = 185 nM T12119 CY42BH 44447607 IC50 = 52 nM T12119 CDJI75 44447616 IC50 = 97 nM T12119 C5RNK0 44476261 IC50 = 150 nM T12119 C01UWF 44540282 IC50 = 370 nM T12119 CWP9Q3 44540283 IC50 = 520 nM T12119 CKCG52 44540374 IC50 = 110 nM T12119 CPFO82 44540469 IC50 = 530 nM T12119 C46HBA 44540470 IC50 = 190 nM T12119 C5NFE6 44540656 IC50 = 710 nM T12119 C2MF7Z 44540754 IC50 = 2200 nM T12119 C5O4TM 44540839 IC50 = 320 nM T12119 CYM71J 44543780 IC50 = 64 nM T12119 CD4LN9 44543781 IC50 = 49 nM T12119 CE0K5T 44543783 IC50 = 350 nM T12119 CS10AL 44543784 IC50 = 350 nM T12119 C17LUC 44543889 IC50 = 260 nM T12119 C9X2SL 44543890 IC50 = 890 nM T12119 CE6HW8 44543891 IC50 = 570 nM T12119 CB83EJ 44544123 IC50 = 430 nM T12119 CN64WQ 44544347 IC50 = 53 nM T12119 CQ79RB 44544349 IC50 = 170 nM T12119 CSV3F9 44544441 IC50 = 1900 nM T12119 C0RI5Z 44544444 IC50 = 550 nM T12119 CK8T7U 44544546 IC50 = 360 nM T12119 C7B0LF 44544548 IC50 = 3100 nM T12119 COJ7H6 44544644 IC50 = 310 nM T12119 CYJB15 44544645 IC50 = 190 nM T12119 CIO82A 44544649 IC50 = 1600 nM T12119 C8RAF0 44544851 IC50 = 230 nM T12119 CWKZ36 44544853 IC50 = 550 nM T12119 C6AX2C 44544950 IC50 = 430 nM T12119 CGB50M 44545053 IC50 = 520 nM T12119 C6VF4T 44545055 IC50 = 4600 nM T12119 CU16DA 44545166 IC50 = 160 nM T12119 C9V7OF 44545167 IC50 = 400 nM T12119 CW78UO 44545168 IC50 = 97 nM T12119 CNZ12F 44545169 IC50 = 51 nM T12119 CCD1V2 44545286 IC50 = 1600 nM T12119 C5KZ2M 44545289 IC50 = 73 nM T12119 C9JK4V 44545402 IC50 = 1700 nM T12119 C6L8QO 44545403 IC50 = 87 nM T12119 CGLQ31 44552634 IC50 = 450 nM T12119 CC2IO4 44552811 IC50 = 1900 nM T12119 CTX13C 44555196 IC50 = 340 nM T12119 CTOP92 44555493 IC50 = 1200 nM T12119 CPM4I9 44555494 IC50 = 620 nM T12119 CNIL25 44555495 IC50 = 710 nM T12119 CB7H1V 44555496 IC50 = 120 nM T12119 CRKJ17 44555497 IC50 = 20 nM T12119 CA51HC 45136898 IC50 = 700 nM T12119 C40BIM 45139151 IC50 = 289 nM T12119 C06OIB 45484762 IC50 = 220 nM T12119 C54WEV 45484834 IC50 = 190 nM T12119 C92VQO 45486749 IC50 = 430 nM T12119 CT6X5N 45486750 IC50 = 480 nM T12119 CUV4N8 45486753 IC50 = 340 nM T12119 CE3QN6 45486773 IC50 = 970 nM T12119 C4KE2L 45486790 IC50 = 1500 nM T12119 CO02YA 45486800 IC50 = 780 nM T12119 C7IJD3 45486807 IC50 = 2500 nM T12119 CJZ4V9 45486818 IC50 = 500 nM T12119 CO3WE7 45487636 IC50 = 450 nM T12119 CBF4V3 45487638 IC50 = 160 nM T12119 C2SBY9 45487649 IC50 = 220 nM T12119 C8S6XW 45487650 IC50 = 580 nM T12119 CUS1O7 45487651 IC50 = 180 nM T12119 C53LZH 45487654 IC50 = 110 nM T12119 C3AS1D 45487655 IC50 = 740 nM T12119 CW6D1P 45487658 IC50 = 84 nM T12119 CI25ZY 45487659 IC50 = 370 nM T12119 CG4E8B 45487661 IC50 = 1700 nM T12119 C8U6FY 45487662 IC50 = 430 nM T12119 CQI8P1 45487664 IC50 = 590 nM T12119 CGO10H 45487665 IC50 = 390 nM T12119 CGTB06 45487669 IC50 = 440 nM T12119 C0QGC7 45487670 IC50 > 5000 nM T12119 CLS42J 45487672 IC50 = 180 nM T12119 C1LSQ2 45487677 IC50 = 380 nM T12119 CW50UZ 45487679 IC50 = 210 nM T12119 CD8G1M 46700763 IC50 = 199.99 nM T12119 CTZ8B1 46832688 IC50 = 30 nM T12119 COS50X 46833288 IC50 > 250 nM T12119 CG6A9H 46840681 IC50 = 49 nM T12119 C91HYQ 46840813 IC50 = 8.999 nM T12119 CSR4H8 46840814 IC50 = 7.8 nM T12119 C0DE7L 46840815 IC50 = 10 nM T12119 CT6W5S 46840816 IC50 = 40 nM T12119 CLU0N8 46840817 IC50 = 7.6 nM T12119 CTNB01 46840818 IC50 = 7.199 nM T12119 CS1T4U 46840947 IC50 = 2.1 nM T12119 C6L7MP 46840948 IC50 = 1.2 nM T12119 C1L0GS 46840949 IC50 = 3.7 nM T12119 C4C0ED 46840950 IC50 = 11 nM T12119 CTYL75 46840951 IC50 = 3.1 nM T12119 COH1P2 46841079 IC50 = 4.8 nM T12119 CLOA87 46841080 IC50 = 4.6 nM T12119 COY73K 46841081 IC50 = 2.1 nM T12119 CT13OG 46841082 IC50 = 4.9 nM T12119 C5YT8R 46841083 IC50 = 8.8 nM T12119 CAH2P5 46841214 IC50 = 52 nM T12119 CSI02O 46841215 IC50 = 1.3 nM T12119 CI1YK3 46841216 IC50 = 13 nM T12119 CROG89 46841217 IC50 = 4.8 nM T12119 CJH48A 46841218 IC50 = 1.2 nM T12119 C5A6KY 46841351 IC50 = 6.2 nM T12119 CV3AK1 46841354 IC50 = 7 nM T12119 CEX70K 46841498 IC50 = 3.8 nM T12119 CD8M3F 46841499 IC50 = 2.6 nM T12119 C3ZVJ7 46841500 IC50 = 5.1 nM T12119 CO76ID 46841501 IC50 = 30 nM T12119 C13LRS 46841502 IC50 = 6.2 nM T12119 C26HOV 46841645 IC50 = 5.8 nM T12119 CE46RS 46841647 IC50 = 4 nM T12119 CS5EJ1 46841648 IC50 = 19 nM T12119 CA06HF 46841786 IC50 = 1.6 nM T12119 CRE97F 46841787 IC50 = 13 nM T12119 COV0Q3 46841788 IC50 = 3.1 nM T12119 C2OWF8 46841789 IC50 = 5 nM T12119 C45AJX 46841790 IC50 = 0.7 nM T12119 CZ7WY4 46841934 IC50 = 29 nM T12119 CQ2E3L 46841935 IC50 = 13 nM T12119 CVL2J1 46841936 IC50 = 3.5 nM T12119 CK46QG 46841937 IC50 = 11 nM T12119 C4PS3C 46841938 IC50 = 3.8 nM T12119 CVC1T9 46842088 IC50 = 12 nM T12119 C3B8XW 46842089 IC50 = 34 nM T12119 CJK53D 46933697 Ki = 340 nM T12119 C8Z0VS 49831248 IC50 = 9 nM T12119 C2VZ5R 49865606 IC50 = 430 nM T12119 C0S8XD 49865953 IC50 = 272 nM T12119 CZT73H 49865954 IC50 = 187 nM T12119 CLW9X4 49866005 Ki = 0.111 nM T12119 CGK7D1 49866006 IC50 = 65 nM T12119 CT8Q4D 49866007 IC50 = 111 nM T12119 C5XM4O 49866055 IC50 = 1368 nM T12119 C9RHZ1 49866056 IC50 = 781 nM T12119 C9KJ3M 49866057 IC50 = 243 nM T12119 CCI6M4 49866115 IC50 = 412 nM T12119 C04DAU 49866116 IC50 = 71 nM T12119 CC5T4F 49866117 IC50 = 41 nM T12119 C6E9ZI 49866118 IC50 = 128 nM T12119 C50GUH 49866119 IC50 = 162 nM T12119 CWS2I4 49866122 IC50 = 1260 nM T12119 CT45VM 49866175 IC50 = 222 nM T12119 C3BI1A 49866176 IC50 = 373 nM T12119 CH59FR 49866206 IC50 = 2770 nM T12119 CC0FA8 49866207 IC50 = 1250 nM T12119 CX82BO 49866244 IC50 = 490 nM T12119 C4MD3J 49869304 IC50 = 6966 nM T12119 CLJ89W 49869305 IC50 = 64 nM T12119 C9YM1Q 49869306 IC50 = 109 nM T12119 CQ9PZ5 49869459 IC50 = 562 nM T12119 C2N0XV 49869747 IC50 = 613 nM T12119 CENW12 50925404 IC50 = 810 nM T12119 CUK75Z 50925405 IC50 = 195 nM T12119 C63UYC 50925406 IC50 = 155 nM T12119 CZ61NW 51333599 IC50 = 43 nM T12119 C06OXV 52920492 IC50 = 14500 nM T12119 C6RFU2 53025800 IC50 = 381 nM T12119 CX0F3U 53025803 IC50 > 3000 nM T12119 C4W9BZ 53025831 IC50 > 3000 nM T12119 CPD0F2 53025889 IC50 = 414 nM T12119 C0GF1R 53025891 IC50 = 48 nM T12119 CMU7X8 53025901 IC50 = 321 nM T12119 C08VWL 53025902 IC50 = 312 nM T12119 CY74FO 53025906 IC50 = 437 nM T12119 C5PB6K 53025909 IC50 = 436 nM T12119 CY3R7J 53058099 IC50 = 280 nM T12119 C8BG5J 53058100 IC50 = 94 nM T12119 C02VSJ 53058119 IC50 = 563 nM T12119 CK59VP 53058205 IC50 = 160 nM T12119 CMS2F7 53239561 IC50 = 3020 nM T12119 CRB6N5 53307604 IC50 = 177.83 nM T12119 CZMA05 53318633 IC50 = 147 nM T12119 CI3LN7 53318774 IC50 = 106 nM T12119 C8JF0H 53319960 IC50 = 64 nM T12119 C61MZW 53320375 IC50 = 132 nM T12119 C2V4UH 53321261 IC50 = 185 nM T12119 CV9BR7 53321262 IC50 = 282 nM T12119 C73HYL 53321263 IC50 = 325 nM T12119 C0QP5Z 53322583 IC50 = 115 nM T12119 C4SMT2 53322584 IC50 = 10 nM T12119 C69OZF 53322585 IC50 = 29 nM T12119 CV8WI6 53322586 IC50 = 715 nM T12119 C0ZS1R 53326494 IC50 = 49 nM T12119 C0AS8V 53326495 IC50 = 477 nM T12119 C7J3AP 53326496 IC50 = 106 nM T12119 CM83SD 53326497 IC50 = 46 nM T12119 C23WVS 53361524 Ki = 35 nM T12119 CRG3B4 53362166 IC50 = 9900 nM T12119 CUV36C 53362167 IC50 > 10000 nM T12119 C3M7ZX 53362168 IC50 = 1400 nM T12119 CL9AP1 53362169 IC50 = 1400 nM T12119 C74RVP 53362170 IC50 = 5000 nM T12119 CI8UK5 53362171 IC50 = 600 nM T12119 CPDG10 53362214 IC50 = 13000 nM T12119 CPLK56 53362438 IC50 > 10000 nM T12119 CNYO17 53362439 IC50 = 3400 nM T12119 C1W3SR 53362440 IC50 = 5000 nM T12119 CUW9Z1 53362441 IC50 = 2600 nM T12119 C6VE8U 53362442 IC50 = 8100 nM T12119 C5TW8P 53362499 IC50 = 1200 nM T12119 C54YUZ 53362500 IC50 = 400 nM T12119 C6CR4I 53362501 IC50 = 900 nM T12119 CJW0B3 53362502 IC50 = 600 nM T12119 CXD49H 53362503 IC50 > 10000 nM T12119 C9YB0C 53362556 IC50 > 10000 nM T12119 C64XGS 53362557 IC50 > 10000 nM T12119 CBAC86 53362558 IC50 = 800 nM T12119 CYX87Q 53362559 IC50 = 300 nM T12119 C9D3FA 53362560 IC50 = 800 nM T12119 CAIL74 53362921 IC50 > 10000 nM T12119 C86LAG 53362922 IC50 > 10000 nM T12119 CGF0X2 53362968 IC50 = 2500 nM T12119 C35ADH 53362970 IC50 > 10000 nM T12119 C09HYM 53362971 IC50 > 10000 nM T12119 C8B1ZY 53362973 IC50 = 1900 nM T12119 COJ14N 53363026 IC50 > 10000 nM T12119 C3F5OH 53363027 IC50 > 10000 nM T12119 CTI0E5 53363028 IC50 > 10000 nM T12119 C3S7ND 53363029 IC50 > 10000 nM T12119 C3NS0D 53363030 IC50 > 10000 nM T12119 CVF6B9 53363031 IC50 > 10000 nM T12119 CM6L7R 53363032 IC50 > 10000 nM T12119 CWA14L 53802926 IC50 = 1000 nM T12119 CH4XK2 54580606 IC50 = 200 nM T12119 CF02UC 54580607 IC50 = 7370 nM T12119 CQP04Y 54580639 IC50 = 1900 nM T12119 C59QAD 54580640 IC50 = 30 nM T12119 C9QK4B 54580641 IC50 > 5000 nM T12119 CHY4B9 54581612 IC50 > 5000 nM T12119 C65ZGC 54581613 IC50 = 40 nM T12119 CZIX38 54581614 IC50 = 60 nM T12119 CB2J8I 54581615 IC50 = 70 nM T12119 CD1JB9 54581652 IC50 = 110 nM T12119 C7QUT0 54581653 IC50 = 1740 nM T12119 CM6Y8G 54582642 IC50 = 630 nM T12119 C8DZC4 54582643 IC50 = 1480 nM T12119 COR31N 54583597 IC50 = 220 nM T12119 C90TRJ 54584552 IC50 = 6080 nM T12119 CMG7X5 54584553 IC50 = 40 nM T12119 CJZ98Y 54584554 IC50 = 60 nM T12119 C9ONC3 54584569 IC50 > 10000 nM T12119 CXSN61 54584585 IC50 = 1100 nM T12119 CBR47V 54584586 IC50 = 1810 nM T12119 C86HBI 54585496 IC50 = 3210 nM T12119 CX0QG3 54585497 IC50 = 6140 nM T12119 C6PT7D 54585524 IC50 = 90 nM T12119 CM12JS 54585525 IC50 = 1630 nM T12119 CF82CK 54586498 IC50 > 5000 nM T12119 CQJV82 54586499 IC50 > 5000 nM T12119 CUT1P3 54587491 IC50 = 1190 nM T12119 CAH0U6 54587492 IC50 = 60 nM T12119 C13UGJ 54587534 IC50 > 5000 nM T12119 C4CV5R 54587535 IC50 > 5000 nM T12119 CI9YU8 56599150 IC50 = 1.1 nM T12119 CG5T6R 56659661 IC50 = 851.14 nM T12119 CUGJ21 56666584 IC50 = 12589.25 nM T12119 C39VWM 56676812 IC50 = 58.88 nM T12119 C2LD6Y 56680137 IC50 = 125.89 nM T12119 C5I4WJ 56680138 IC50 = 1230.27 nM T12119 CN5SE7 56683480 IC50 = 3630.78 nM T12119 C15EFA 56961983 IC50 = 237 nM T12119 C3TMW0 56961984 IC50 = 188 nM T12119 C7PE9X 56961986 IC50 = 291 nM T12119 CO3D7N 56962034 IC50 = 177 nM T12119 CRN8T7 56962087 IC50 = 98.3 nM T12119 CQT5I3 57328465 IC50 = 240 nM T12119 CS1XE6 57328466 IC50 = 110 nM T12119 CA64TK 57389500 IC50 = 9700 nM T12119 C67NZF 57390663 IC50 > 30000 nM T12119 CDKJ90 57394169 IC50 > 30000 nM T12119 CZ3FJ9 57395950 IC50 > 30000 nM T12119 CBR80E 57404708 IC50 = 96 nM T12119 CFC34T 57405056 IC50 = 110 nM T12119 CBFD09 57405219 Ki = 19 nM T12119 CLQ04N 57405559 Ki = 113 nM T12119 CRBD24 57405732 IC50 = 74 nM T12119 CJNA87 57406788 IC50 = 140 nM T12119 CT54IO 57407169 IC50 = 42 nM T12119 CUM1G7 57407346 IC50 = 64 nM T12119 CYO3K6 57407347 Ki = 59 nM T12119 COUZ63 57494822 IC50 = 2 nM T12119 C5ST6N 57494823 IC50 = 5.4 nM T12119 C51MWI 57494824 IC50 = 15 nM T12119 CHU68T 57494825 IC50 = 38 nM T12119 CCJ93I 57494826 IC50 = 4.1 nM T12119 CR34CL 57582353 IC50 = 36000 nM T12119 CU1R0H 57779770 IC50 = 254 nM T12119 CL1NR8 57779793 IC50 = 359 nM T12119 CCYG05 59263528 IC50 = 60 nM T12119 C45DCP 59352142 IC50 = 270 nM T12119 C6HE7J 59352158 IC50 = 8 nM T12119 CWXM63 59352188 IC50 > 1000 nM T12119 CI9N1Q 59352252 IC50 = 150 nM T12119 CI8O4J 59352254 IC50 = 230 nM T12119 CL4M9F 59352317 IC50 = 190 nM T12119 CXG8W3 59352369 IC50 = 430 nM T12119 C6RKA8 59352665 IC50 = 10 nM T12119 CT7S3U 59352762 IC50 = 110 nM T12119 C0EU4H 59352764 IC50 = 1150 nM T12119 CA4MY8 59436470 IC50 = 70 nM T12119 CE8AZ3 59436502 IC50 = 3.7 nM T12119 CYPZ53 59436514 IC50 = 1710.02 nM T12119 CSD03G 59436531 IC50 = 89.99 nM T12119 CVE08F 59436540 IC50 = 2320.06 nM T12119 C9J7FB 59436552 IC50 = 3.8 nM T12119 C0SB9O 59436554 IC50 = 10000 nM T12119 CXHO91 59436576 IC50 = 24940.2 nM T12119 C2BH6M 59436587 IC50 = 70 nM T12119 C9LKX1 59436588 IC50 = 12540.07 nM T12119 CQ9MV4 59436597 IC50 = 810.03 nM T12119 CF27SW 59436599 IC50 = 10 nM T12119 CI21SG 59436612 IC50 = 10000 nM T12119 C59ADR 59436616 IC50 = 3769.64 nM T12119 C92MKJ 59436623 IC50 = 100 nM T12119 CYF3R7 60167367 IC50 = 26000 nM T12119 CDVX75 60199269 IC50 < 2000 nM T12119 CSA3I9 60200914 IC50 = 680 nM T12119 CK76WB 60200915 IC50 > 11000 nM T12119 CI40XK 60201083 IC50 = 420 nM T12119 CNR41U 60201084 IC50 = 750 nM T12119 CO5HD0 60201085 IC50 = 160 nM T12119 CA57OQ 60201086 IC50 = 18000 nM T12119 C5UKQ8 60201087 IC50 = 21000 nM T12119 CA7NI3 60201088 IC50 = 780 nM T12119 C56KOS 60201255 IC50 = 140 nM T12119 C1YQ8J 60201256 IC50 = 990 nM T12119 CVW28G 60201257 IC50 = 140 nM T12119 CC82DM 65459349 IC50 = 7000 nM T12119 C6EJ3F 66551245 IC50 = 251.19 nM T12119 COTD35 66667669 IC50 = 76 nM T12119 CD2HV3 66813354 IC50 = 3162.28 nM T12119 C78XLS 66813470 IC50 = 158.49 nM T12119 CAOB97 66813557 IC50 = 100 nM T12119 C89WUE 66813671 IC50 = 79.43 nM T12119 CSY3F6 66813695 IC50 = 3981.07 nM T12119 CPK67V 66813703 IC50 = 1258.93 nM T12119 C7DX6Z 66813839 IC50 = 63.1 nM T12119 CH2D5F 66813859 IC50 = 79.43 nM T12119 C90OSR 66813870 IC50 = 158.49 nM T12119 COZ0U9 66813914 IC50 = 79.43 nM T12119 C5OTD2 66813927 IC50 = 100 nM T12119 C39PEZ 66814019 IC50 = 398.11 nM T12119 CG80RS 66814110 IC50 = 251.19 nM T12119 CCG8F3 66905459 IC50 = 2999.85 nM T12119 C56SKG 66978520 IC50 = 151 nM T12119 CD32LX 67461417 IC50 = 50 nM T12119 CBQ5O1 67523614 IC50 = 81 nM T12119 CM7AT3 67523656 IC50 = 35 nM T12119 C3U7IX 67981754 Ki = 25 nM T12119 CDL0E8 67981901 Ki = 75 nM T12119 C65EUW 68109680 IC50 = 130 nM T12119 CFGE17 68153368 IC50 < 2000 nM T12119 CGE3W8 68657852 IC50 = 10000 nM T12119 CT1YQ7 68680505 IC50 = 6900 nM T12119 C52LVB 68710093 IC50 = 20 nM T12119 CBH6T3 69003776 IC50 = 1000 nM T12119 CXF5P9 69213151 IC50 = 1995.26 nM T12119 COF9A2 70355061 IC50 = 8 nM T12119 CZ39KM 70681034 IC50 = 13500 nM T12119 C1N4OJ 70681038 IC50 = 8800 nM T12119 CG9B0S 70681039 IC50 = 5700 nM T12119 CP8XS4 70681040 IC50 = 1800 nM T12119 C4Z9CP 70681041 IC50 > 30000 nM T12119 CC7Q1P 70681042 IC50 = 10800 nM T12119 CF85AB 70681063 IC50 = 80 nM T12119 C9LW7K 70681064 IC50 = 20 nM T12119 CX6UZ8 70681066 IC50 = 1400 nM T12119 CHP32B 70681067 IC50 = 6500 nM T12119 CS8V7G 70681068 IC50 = 190 nM T12119 C1KL9H 70681069 IC50 = 5150 nM T12119 CL28PN 70682458 IC50 = 794.33 nM T12119 CJV64I 70683156 IC50 = 2900 nM T12119 CU73VN 70683159 IC50 = 6100 nM T12119 CD7U5Y 70683160 IC50 = 7300 nM T12119 C9BR3A 70683161 IC50 = 620 nM T12119 CT6NB4 70683162 IC50 = 5900 nM T12119 C3RC0E 70683163 IC50 = 11100 nM T12119 C36DYJ 70683164 IC50 = 2300 nM T12119 CN79ZX 70683165 IC50 = 1200 nM T12119 C1D5SA 70683166 IC50 = 25700 nM T12119 CRXZ90 70683167 IC50 = 1300 nM T12119 C94GTH 70683168 IC50 = 260 nM T12119 C3ZY6F 70683178 IC50 = 50 nM T12119 C7NAV4 70683180 IC50 = 310 nM T12119 CN17AS 70683181 IC50 = 140 nM T12119 CA8VC6 70683182 IC50 = 100 nM T12119 C7RU0T 70683183 IC50 > 30000 nM T12119 C6QC5J 70683184 IC50 = 30 nM T12119 C3P0LX 70683185 IC50 = 4600 nM T12119 CLG7N8 70683186 IC50 = 9600 nM T12119 CK6JM8 70683187 IC50 = 300 nM T12119 CWK3H8 70683188 IC50 = 510 nM T12119 C1ARO8 70684544 IC50 = 501.19 nM T12119 C3T1WM 70684545 IC50 = 25118.86 nM T12119 C4I0ZH 70684546 IC50 > 10000 nM T12119 CUX59H 70685234 IC50 > 10000 nM T12119 CIV4S6 70685239 IC50 = 2000 nM T12119 CEV37L 70685240 IC50 = 5300 nM T12119 CL7Q3D 70685241 IC50 = 11300 nM T12119 C48GHD 70685242 IC50 = 9800 nM T12119 CFV0A8 70685243 IC50 > 30000 nM T12119 CLIN14 70685244 IC50 = 3900 nM T12119 CLW68N 70685259 IC50 = 60 nM T12119 C65PTC 70685263 IC50 = 830 nM T12119 C2IDQ6 70685264 IC50 = 20 nM T12119 C02FWG 70685265 IC50 = 50 nM T12119 CO1ZR5 70685266 IC50 = 130 nM T12119 C9BA4Z 70685268 IC50 = 14000 nM T12119 CRP7Z1 70685269 IC50 = 1130 nM T12119 CRDJ83 70686683 IC50 = 501.19 nM T12119 CI0Z9V 70687389 IC50 = 3100 nM T12119 CEAK85 70687392 IC50 = 1800 nM T12119 CC32TO 70687393 IC50 = 500 nM T12119 CE7M6D 70687413 IC50 = 7200 nM T12119 CC3UR7 70687414 IC50 = 6600 nM T12119 C3E9VJ 70687415 IC50 = 120 nM T12119 C5I4WO 70687416 IC50 = 7620 nM T12119 CQ29WE 70687417 IC50 = 3810 nM T12119 C0A3VH 70687418 IC50 = 160 nM T12119 CD2EW1 70688785 IC50 = 125.89 nM T12119 CH7Z3Q 70689449 IC50 > 10000 nM T12119 C4QY7T 70689451 IC50 > 30000 nM T12119 C6YJL1 70689452 IC50 = 440 nM T12119 CALX60 70689470 IC50 = 3510 nM T12119 C13OAI 70689471 IC50 = 25200 nM T12119 C1QX5M 70689472 IC50 = 3260 nM T12119 CO89VX 70689473 IC50 = 1100 nM T12119 C56TAW 70689474 IC50 = 2700 nM T12119 CM3PD8 70689475 IC50 = 950 nM T12119 CV82BX 70690866 IC50 = 794.33 nM T12119 C8R0SZ 70691558 IC50 = 1600 nM T12119 CRXG05 70691559 IC50 = 2000 nM T12119 CYJ3F6 70691560 IC50 = 900 nM T12119 CK6I2V 70691577 IC50 = 40 nM T12119 C7ET5J 70691581 IC50 = 2290 nM T12119 CJ85NC 70691582 IC50 = 70 nM T12119 C27IPY 70691584 IC50 = 180 nM T12119 C8OKQ0 70693647 IC50 = 3200 nM T12119 CLN9F4 70693648 IC50 = 1300 nM T12119 CM3LU4 70693649 IC50 = 880 nM T12119 C3GVN0 70693667 IC50 = 260 nM T12119 CKP02Q 70693669 IC50 = 70 nM T12119 C6N3DT 70693670 IC50 = 2900 nM T12119 CB0I5R 70693671 IC50 = 4700 nM T12119 CEI84H 70693672 IC50 = 270 nM T12119 C6GCU1 70693673 IC50 = 40 nM T12119 CHUE45 70693674 IC50 = 30 nM T12119 CCQ49A 70695045 IC50 = 630.96 nM T12119 CBCD89 70695046 IC50 = 794.33 nM T12119 C63MTE 70695047 IC50 = 79.43 nM T12119 CEK60M 70695761 IC50 = 440 nM T12119 C1AUW5 70695763 IC50 = 5500 nM T12119 CX6L3G 70695764 IC50 = 1500 nM T12119 CF4HZ3 70695774 IC50 = 150 nM T12119 C7H2ER 70695778 IC50 > 30000 nM T12119 CBHD70 70695780 IC50 = 40 nM T12119 C7G1UY 70695781 IC50 = 3490 nM T12119 CZL9G2 70695782 IC50 = 20 nM T12119 CKCE67 70695783 IC50 = 1700 nM T12119 CUL37Y 70695784 IC50 = 330 nM T12119 C26OHM 70695785 IC50 = 40 nM T12119 CD1V2W 70695786 IC50 = 60 nM T12119 CE9W1Z 70814180 IC50 = 1500 nM T12119 C7Z6HJ 70814238 IC50 = 404 nM T12119 C7JD8A 70814244 IC50 = 344 nM T12119 C1ST3M 70814308 IC50 = 311 nM T12119 C5OT1G 70814333 IC50 = 478 nM T12119 C51SEO 70866438 IC50 = 11 nM T12119 C2FNI6 71259239 IC50 = 38 nM T12119 CG0L7O 71259621 IC50 = 120 nM T12119 CJA92P 71290100 Ki = 16 nM T12119 CR4L9T 71449282 IC50 = 125.89 nM T12119 CHF08N 71449283 IC50 = 25.12 nM T12119 CMB7U1 71449284 IC50 = 398.11 nM T12119 CVY54C 71449294 IC50 > 10000 nM T12119 C7L6QZ 71449295 IC50 > 10000 nM T12119 CIFE14 71451076 IC50 = 63.1 nM T12119 CLSQ82 71451077 IC50 = 398.11 nM T12119 C0RL3C 71451078 IC50 = 31.62 nM T12119 CGJ7K0 71451084 IC50 = 630.96 nM T12119 CI0B8V 71451085 IC50 = 125.89 nM T12119 CXT57R 71452899 IC50 = 39.81 nM T12119 CG21NF 71452900 IC50 = 1995.26 nM T12119 C7D9SN 71452907 IC50 > 10000 nM T12119 C5WU8L 71454670 IC50 = 31.62 nM T12119 C7XQZ4 71454678 IC50 = 39.81 nM T12119 CVU2O8 71454679 IC50 > 10000 nM T12119 C1X6TY 71456401 IC50 = 25.12 nM T12119 C7AL1C 71456402 IC50 = 100 nM T12119 CORH12 71456403 IC50 = 251.19 nM T12119 C9FX5O 71456404 IC50 = 6309.57 nM T12119 CR4ZO3 71456412 IC50 = 31.62 nM T12119 CC3Q9J 71456413 IC50 = 25.12 nM T12119 C7OW1B 71458245 IC50 > 10000 nM T12119 CIKE31 71458259 IC50 = 199.53 nM T12119 C6K4BO 71460096 IC50 = 1000 nM T12119 C9A7HP 71460097 IC50 = 3162.28 nM T12119 CYBR37 71460098 IC50 = 63.1 nM T12119 CQW3L4 71460099 IC50 > 10000 nM T12119 CSB76D 71460108 IC50 = 50.12 nM T12119 CT7KJ9 71460109 IC50 = 1000 nM T12119 CQ30OU 71461829 IC50 > 10000 nM T12119 CV7ML5 71461830 IC50 = 199.53 nM T12119 C2MC6B 71522734 IC50 = 0.3 nM T12119 CM1B0W 71523649 IC50 = 24000 nM T12119 CHAU76 71555980 IC50 = 486 nM T12119 C25YAP 71555982 IC50 = 190 nM T12119 C0AO1Y 71556159 IC50 = 21 nM T12119 CF10XG 71556345 IC50 = 4 nM T12119 CL94JM 71556743 IC50 = 74 nM T12119 C1DH3U 71556801 IC50 = 244 nM T12119 C3EC1H 71557026 IC50 = 1.7 nM T12119 CL85YK 71557177 IC50 = 5.3 nM T12119 CY59CA 71557630 IC50 = 1.1 nM T12119 CTI52S 71557789 IC50 = 4 nM T12119 CO09GI 71558118 IC50 = 2.6 nM T12119 CMKH30 71558122 IC50 = 11 nM T12119 C2SP3F 71558162 IC50 = 8.7 nM T12119 C48RIB 71558271 IC50 = 6.8 nM T12119 CEJR19 71558272 IC50 = 237 nM T12119 CK2HF0 71558274 IC50 = 51 nM T12119 CU5L4F 71558467 IC50 = 3 nM T12119 CUI6M5 71558468 IC50 = 3.6 nM T12119 C0DO9Y 71558578 IC50 = 3.3 nM T12119 CS8M1O 71558621 IC50 = 4.4 nM T12119 C2ZN4G 71558725 IC50 = 331 nM T12119 CIDS01 71558883 IC50 = 0.9 nM T12119 CY6Z1T 71558917 IC50 = 0.5 nM T12119 CHRO29 71558920 IC50 = 1.7 nM T12119 C9WGA1 71559034 IC50 = 13 nM T12119 CE60JF 71559072 IC50 = 1.7 nM T12119 CA8GW3 71559220 IC50 = 51 nM T12119 C20ELR 71559363 IC50 = 222 nM T12119 C2W5PU 71559364 IC50 = 2300 nM T12119 CJXK67 71559365 IC50 = 0.4 nM T12119 CYU36D 71566103 IC50 = 872 nM T12119 C76IAH 71577327 IC50 = 470 nM T12119 C8XIJ2 71582572 IC50 = 90 nM T12119 C02MBD 71582575 IC50 = 14 nM T12119 C1Y9SA 71583000 IC50 = 3162.28 nM T12119 CLAZ62 71585735 IC50 = 120 nM T12119 CRC01X 71585929 IC50 = 48 nM T12119 CXA29H 71585930 IC50 = 51 nM T12119 CPI61F 71586033 IC50 = 510 nM T12119 C4U3GM 71586128 IC50 = 30 nM T12119 CNY52I 71586326 IC50 = 590 nM T12119 C8Z6JV 71612390 IC50 = 35 nM T12119 CE54ZC 71616019 IC50 = 240 nM T12119 CE8FD1 71626223 IC50 = 251.19 nM T12119 CK0NE8 71654730 IC50 = 264 nM T12119 CEKY57 71654731 IC50 = 260 nM T12119 CT08ZN 71654732 IC50 = 103 nM T12119 C1F4AB 71654733 IC50 = 443 nM T12119 CSF4A6 71654807 IC50 = 229 nM T12119 CXS37M 71654810 IC50 = 85 nM T12119 CVH4T5 71655778 IC50 = 181 nM T12119 CD5IO2 71655779 IC50 = 67 nM T12119 CV54NY 71666500 IC50 < 2000 nM T12119 C5LM0G 71711363 IC50 = 390 nM T12119 CGOV74 71711365 IC50 = 9200 nM T12119 C1VC7P 71711696 IC50 = 460 nM T12119 C6HWZ5 71711765 IC50 = 2600 nM T12119 C8D7FJ 71711834 IC50 = 38.6 nM T12119 CD4Z0Y 71711979 IC50 = 37 nM T12119 CV2X6E 71712184 IC50 = 21 nM T12119 CK0L1B 71712241 IC50 = 30 nM T12119 C7N1DW 71716173 IC50 = 920.03 nM T12119 C8Y7HN 71716174 IC50 = 930.04 nM T12119 C3J1XH 71716175 IC50 = 979.94 nM T12119 CE8XA3 71716176 IC50 = 1000 nM T12119 C07HQC 71716177 IC50 = 1000 nM T12119 CAMB96 71716178 IC50 = 1000 nM T12119 C82MYH 71716179 IC50 = 759.98 nM T12119 C61KFL 71716180 IC50 = 780.01 nM T12119 CM7E3O 71716181 IC50 = 840.04 nM T12119 C39UCK 71716184 IC50 = 899.91 nM T12119 CSE98K 71716185 IC50 = 600.07 nM T12119 CQBU61 71716186 IC50 = 659.93 nM T12119 CK5DM4 71716187 IC50 = 670.04 nM T12119 CKPD58 71716188 IC50 = 739.95 nM T12119 CI5G4O 71716189 IC50 = 430.03 nM T12119 CGRA37 71716190 IC50 = 470 nM T12119 C53ZTP 71716191 IC50 = 479.95 nM T12119 CP7YB8 71716192 IC50 = 520 nM T12119 CAK0F9 71716197 IC50 = 540.01 nM T12119 CH5RM2 71716198 IC50 = 340.02 nM T12119 CCP0O5 71716199 IC50 = 340.02 nM T12119 CBHG02 71716200 IC50 = 419.95 nM T12119 CI2C7D 71716201 IC50 = 419.95 nM T12119 CO6D0I 71716202 IC50 = 299.99 nM T12119 CS0W3O 71716203 IC50 = 299.99 nM T12119 CPKA91 71716209 IC50 = 299.99 nM T12119 CH1AE2 71716210 IC50 = 329.99 nM T12119 CJC1L6 71716211 IC50 = 229.99 nM T12119 CL20KF 71716212 IC50 = 229.99 nM T12119 CG0R2P 71716218 IC50 = 199.99 nM T12119 C8TH5A 71716219 IC50 = 129.99 nM T12119 C4BP7F 71716220 IC50 = 129.99 nM T12119 CR7Z1N 71716221 IC50 = 139.99 nM T12119 CSO95R 71716222 IC50 = 139.99 nM T12119 CMQ90P 71716223 IC50 = 159.99 nM T12119 C90NWB 71716229 IC50 = 100 nM T12119 CU56WA 71716230 IC50 = 110 nM T12119 CS61ZB 71716231 IC50 = 110 nM T12119 CV85ME 71716232 IC50 = 110 nM T12119 CW4G5R 71716233 IC50 = 120.01 nM T12119 CH5VT7 71716234 IC50 = 80 nM T12119 CN5L0B 71716243 IC50 = 97.01 nM T12119 C7HE9C 71716244 IC50 = 60.01 nM T12119 CMOS25 71716245 IC50 = 68.99 nM T12119 CWA3Z5 71716246 IC50 = 78 nM T12119 CPI0W8 71716247 IC50 = 40 nM T12119 CWH60K 71716248 IC50 = 40 nM T12119 C4LN9C 71716249 IC50 = 41 nM T12119 CO0T7W 71716250 IC50 = 44 nM T12119 CYMF78 71716251 IC50 = 50 nM T12119 CYX48P 71716252 IC50 = 50 nM T12119 C5FBJ9 71716259 IC50 = 50 nM T12119 C0Z4FN 71716260 IC50 = 53 nM T12119 CZ1US8 71716261 IC50 = 56 nM T12119 CZ5PL8 71716262 IC50 = 57 nM T12119 C9LQM7 71716263 IC50 = 34 nM T12119 C52GAC 71716264 IC50 = 25 nM T12119 CI4TQ3 71716265 IC50 = 25 nM T12119 C9OFK3 71716266 IC50 = 25 nM T12119 CVZ1J9 71716267 IC50 = 29 nM T12119 CV3BI9 71716268 IC50 = 18 nM T12119 CQGV74 71716269 IC50 = 20 nM T12119 CI1S2B 71716270 IC50 = 22 nM T12119 CAO4N9 71716271 IC50 = 13 nM T12119 C8CU3A 71716275 IC50 = 15 nM T12119 C31BYG 71716276 IC50 = 14 nM T12119 C1IZ3U 71716277 IC50 = 17 nM T12119 CY6UF2 71716278 IC50 = 9.899 nM T12119 C61MZY 71716280 IC50 = 38895.56 nM T12119 CJM03A 71716281 IC50 = 13999.1 nM T12119 CCQ76M 71716282 IC50 = 17278.26 nM T12119 CO14US 71716283 IC50 = 10000 nM T12119 CB94QY 71716284 IC50 = 10000 nM T12119 C9UY7H 71716285 IC50 = 11000.19 nM T12119 CD7EN4 71716286 IC50 = 12209.56 nM T12119 CN64TS 71716287 IC50 = 5.3 nM T12119 CLD79A 71716288 IC50 = 5.8 nM T12119 C0W5ZA 71716289 IC50 = 7.501 nM T12119 C0ZGL6 71716290 IC50 = 3.9 nM T12119 CV3L1C 71716291 IC50 = 4.4 nM T12119 CMI2B1 71716292 IC50 = 4.4 nM T12119 C9GR2E 71716293 IC50 = 4.5 nM T12119 CDB10L 71716294 IC50 = 4.8 nM T12119 CD8U1P 71716301 IC50 = 9421.06 nM T12119 CCS8R5 71716302 IC50 = 3800.14 nM T12119 CNK16F 71716303 IC50 = 4219.88 nM T12119 C9ND2E 71716304 IC50 = 4540.46 nM T12119 C3HGN9 71716305 IC50 = 5000.35 nM T12119 CSV2C4 71716306 IC50 = 5100.35 nM T12119 C42POI 71716307 IC50 = 5739.84 nM T12119 CJLI05 71716308 IC50 = 5930.62 nM T12119 CQM6Z4 71716309 IC50 = 1.6 nM T12119 CS6W0U 71716310 IC50 = 2.1 nM T12119 CU2OE8 71716311 IC50 = 2.1 nM T12119 CYL49M 71716312 IC50 = 2.5 nM T12119 C03UZJ 71716313 IC50 = 3.5 nM T12119 C57PCJ 71716314 IC50 = 0.8 nM T12119 C12ZDW 71716316 IC50 = 3339.64 nM T12119 C8JDU6 71716317 IC50 = 2619.99 nM T12119 CQ0EB1 71716318 IC50 = 2700.23 nM T12119 CR4YB3 71716319 IC50 = 2789.97 nM T12119 CTB0P2 71716320 IC50 = 2800.27 nM T12119 C0GK7X 71716322 IC50 = 2470.02 nM T12119 C6CP0L 71716323 IC50 = 1900.2 nM T12119 CG2W1E 71716324 IC50 = 1999.86 nM T12119 CVA4T5 71716329 IC50 = 2099.91 nM T12119 C90RKN 71716330 IC50 = 1669.94 nM T12119 C4ZJB8 71716331 IC50 = 1000 nM T12119 C9FD5V 71716332 IC50 = 1000 nM T12119 C94LAH 71716333 IC50 = 1000 nM T12119 C4PDA6 71716334 IC50 = 1029.91 nM T12119 C4MI8E 71716340 IC50 = 1200.05 nM T12119 C3T8HW 71716341 IC50 = 1200.05 nM T12119 CM4S2N 71716342 IC50 = 1229.99 nM T12119 C74QSF 71716343 IC50 = 1000 nM T12119 CE68JP 71716344 IC50 = 1000 nM T12119 CB32UL 71716345 IC50 = 1000 nM T12119 CV2Y5L 71716788 IC50 = 1000 nM T12119 C4H9GM 71716789 IC50 = 1000 nM T12119 C29SOC 71716790 IC50 = 780.01 nM T12119 C1GJ8P 71716791 IC50 = 780.01 nM T12119 CQ1LS5 71716792 IC50 = 890.02 nM T12119 C41WNH 71716800 IC50 = 909.91 nM T12119 CYK2U9 71716801 IC50 = 550.05 nM T12119 CA9S1X 71716802 IC50 = 579.96 nM T12119 C3JU7Z 71716803 IC50 = 600.07 nM T12119 CDWS76 71716804 IC50 = 620.01 nM T12119 CRJ47Q 71716805 IC50 = 670.04 nM T12119 C0R9BE 71716806 IC50 = 710.07 nM T12119 CUC9M8 71716807 IC50 = 510.04 nM T12119 CF2ZB3 71716813 IC50 = 370 nM T12119 CTS5G4 71716814 IC50 = 380.01 nM T12119 CUSE25 71716815 IC50 = 280.03 nM T12119 CD1TI5 71716816 IC50 = 280.03 nM T12119 C98MHB 71716818 IC50 = 299.99 nM T12119 CYN43M 71716819 IC50 = 310.03 nM T12119 C3CVS1 71716820 IC50 = 310.03 nM T12119 CC4A3K 71716821 IC50 = 319.96 nM T12119 CGO2K5 71716822 IC50 = 229.99 nM T12119 C2FC6A 71716823 IC50 = 229.99 nM T12119 C61LBJ 71716824 IC50 = 239.99 nM T12119 C7EG3T 71716825 IC50 = 239.99 nM T12119 C2QS9F 71716826 IC50 = 169.98 nM T12119 C48SVY 71716831 IC50 = 169.98 nM T12119 C89YVO 71716832 IC50 = 169.98 nM T12119 CWT4X5 71716833 IC50 = 180.01 nM T12119 C7UV9A 71716834 IC50 = 129.99 nM T12119 C3EWQ4 71716835 IC50 = 139.99 nM T12119 CZ29UC 71716838 IC50 = 100 nM T12119 C91PEG 71716839 IC50 = 88 nM T12119 CJU86T 71716840 IC50 = 88 nM T12119 CJ0A3Z 71716844 IC50 = 89.99 nM T12119 CGE5V2 71716845 IC50 = 89.99 nM T12119 CF57SR 71716846 IC50 = 73 nM T12119 CAY75W 71716852 IC50 = 50 nM T12119 CU3W4X 71716853 IC50 = 50 nM T12119 C2PS1A 71716854 IC50 = 52 nM T12119 CKVN89 71716855 IC50 = 32 nM T12119 C9MUK3 71716856 IC50 = 31 nM T12119 CVO98F 71716857 IC50 = 40 nM T12119 C71NCI 71716858 IC50 = 23 nM T12119 CV23HK 71716859 IC50 = 25 nM T12119 C2WLX6 71716860 IC50 = 25 nM T12119 CVE8A0 71716864 IC50 = 18 nM T12119 CBC20I 71716865 IC50 = 18 nM T12119 CUG2V3 71716866 IC50 = 20 nM T12119 C50VRD 71716870 IC50 = 32322.13 nM T12119 CQH2K8 71716871 IC50 = 16 nM T12119 CW1P4H 71716872 IC50 = 8.5 nM T12119 CIZ40M 71716873 IC50 = 9.701 nM T12119 CAB1K8 71716874 IC50 = 37187.76 nM T12119 CP1VN0 71716875 IC50 = 13931.57 nM T12119 C16FMX 71716876 IC50 = 15531.02 nM T12119 C06MXC 71716877 IC50 = 17668.51 nM T12119 CK3WT1 71716878 IC50 = 21998.85 nM T12119 CW8ZO1 71716879 IC50 = 23999.38 nM T12119 CQ95EH 71716880 IC50 = 10869.26 nM T12119 C1NIV7 71716881 IC50 = 11489.47 nM T12119 C2U4DC 71716882 IC50 = 5.8 nM T12119 C5DYO8 71716883 IC50 = 5.8 nM T12119 C7UPM2 71716884 IC50 = 6.899 nM T12119 CKRV13 71716885 IC50 = 7.8 nM T12119 CHGS93 71716886 IC50 = 7.9 nM T12119 C1EIV0 71716887 IC50 = 3.6 nM T12119 CRQB34 71716888 IC50 = 4 nM T12119 C43KCM 71716900 IC50 = 10000 nM T12119 CI2FZ3 71716901 IC50 = 10000 nM T12119 CPI5L2 71716902 IC50 = 10000 nM T12119 C9LM7A 71716903 IC50 = 10000 nM T12119 CSC2Y5 71716904 IC50 = 6899.22 nM T12119 CW3KU8 71716905 IC50 = 4.9 nM T12119 CC3RQ7 71716906 IC50 = 1.7 nM T12119 CWR0C1 71716907 IC50 = 2.1 nM T12119 C93PST 71716908 IC50 = 2.8 nM T12119 CQC9F3 71716909 IC50 = 3.2 nM T12119 CQ87DL 71716910 IC50 = 0.8999 nM T12119 C32QPK 71716911 IC50 = 1.4 nM T12119 CRGT51 71716914 IC50 = 2999.85 nM T12119 CA45CL 71716915 IC50 = 3100.27 nM T12119 CY0QT6 71716916 IC50 = 3110.28 nM T12119 CD0Y9B 71716917 IC50 = 2669.93 nM T12119 CB3I4R 71716918 IC50 = 2900.01 nM T12119 C4NZ8D 71716920 IC50 = 2999.85 nM T12119 C0VHS2 71716921 IC50 = 2180.22 nM T12119 CED4F0 71716922 IC50 = 2399.94 nM T12119 CETC69 71716923 IC50 = 2499.77 nM T12119 CJ5MY8 71716924 IC50 = 1800.11 nM T12119 CR07EV 71716925 IC50 = 1880.18 nM T12119 CM67QB 71716926 IC50 = 1999.86 nM T12119 C76RGV 71716932 IC50 = 1999.86 nM T12119 C8T1WV 71716933 IC50 = 1299.87 nM T12119 C7GA8J 71716934 IC50 = 1500.03 nM T12119 C1OW6J 71716935 IC50 = 1510.08 nM T12119 CAZ9U0 71716936 IC50 = 1599.93 nM T12119 C26NZC 71716937 IC50 = 1020 nM T12119 CX1C4E 71716945 IC50 = 1100.02 nM T12119 CS4V9I 71716946 IC50 = 1100.02 nM T12119 CY62KZ 71716947 IC50 = 1150.01 nM T12119 CM2T3Z 71716948 IC50 = 1000 nM T12119 CLI09J 71716949 IC50 = 1000 nM T12119 C1RXM7 71716950 IC50 = 1000 nM T12119 CDTB07 71717403 IC50 = 930.04 nM T12119 CSI8X3 71717404 IC50 = 960.06 nM T12119 C1L5AX 71717405 IC50 = 1000 nM T12119 CIFD43 71717406 IC50 = 1000 nM T12119 CJ0QH5 71717407 IC50 = 770.02 nM T12119 CLH23X 71717408 IC50 = 770.02 nM T12119 CE65AC 71717409 IC50 = 780.01 nM T12119 CTO6H1 71717410 IC50 = 819.97 nM T12119 C7LKH6 71717415 IC50 = 659.93 nM T12119 C6US5N 71717416 IC50 = 739.95 nM T12119 CDN90U 71717417 IC50 = 449.99 nM T12119 CEGF05 71717418 IC50 = 449.99 nM T12119 C1GIW5 71717419 IC50 = 470 nM T12119 CX2GA8 71717420 IC50 = 470 nM T12119 C2E0GZ 71717421 IC50 = 490 nM T12119 CG4HM6 71717427 IC50 = 530.03 nM T12119 C7X2EC 71717428 IC50 = 370 nM T12119 CKE28S 71717429 IC50 = 380.01 nM T12119 C1WI5O 71717430 IC50 = 380.01 nM T12119 CZ3U4J 71717431 IC50 = 400.04 nM T12119 C9BQT2 71717432 IC50 = 270.02 nM T12119 CR0F1X 71717433 IC50 = 270.02 nM T12119 C1QL6R 71717434 IC50 = 299.99 nM T12119 C3E0YZ 71717439 IC50 = 299.99 nM T12119 CVO89U 71717440 IC50 = 299.99 nM T12119 C1X2GB 71717441 IC50 = 299.99 nM T12119 CHO2P0 71717442 IC50 = 319.96 nM T12119 C7DZC9 71717443 IC50 = 329.99 nM T12119 CLV80P 71717444 IC50 = 219.99 nM T12119 C0G5HM 71717445 IC50 = 249.98 nM T12119 CTY94H 71717446 IC50 = 249.98 nM T12119 CBLJ42 71717450 IC50 = 180.01 nM T12119 C9BXC7 71717451 IC50 = 190.02 nM T12119 C23QOI 71717452 IC50 = 190.02 nM T12119 C26ZUG 71717453 IC50 = 190.02 nM T12119 C8RJ2O 71717454 IC50 = 209.99 nM T12119 CLI05M 71717455 IC50 = 209.99 nM T12119 C8BX3R 71717456 IC50 = 129.99 nM T12119 CGT59N 71717457 IC50 = 129.99 nM T12119 CT0WC6 71717458 IC50 = 129.99 nM T12119 C6G3RZ 71717459 IC50 = 139.99 nM T12119 C5SB9Z 71717463 IC50 = 100 nM T12119 CB6NW5 71717464 IC50 = 110 nM T12119 CODP68 71717465 IC50 = 110 nM T12119 CWZ96L 71717466 IC50 = 120.01 nM T12119 C7SF1O 71717478 IC50 = 90.99 nM T12119 CU29SZ 71717479 IC50 = 93 nM T12119 CXPZ05 71717480 IC50 = 94.99 nM T12119 CW82JH 71717481 IC50 = 98.99 nM T12119 CT85OD 71717482 IC50 = 100 nM T12119 CD0LJ3 71717483 IC50 = 67 nM T12119 C4GVC0 71717484 IC50 = 71.99 nM T12119 CQK4H3 71717485 IC50 = 44 nM T12119 C7I3TV 71717491 IC50 = 53 nM T12119 CC78DL 71717492 IC50 = 30 nM T12119 CC7X2N 71717493 IC50 = 31 nM T12119 C4XYN9 71717494 IC50 = 26 nM T12119 CA5E4Z 71717495 IC50 = 34 nM T12119 CCF83M 71717496 IC50 = 25 nM T12119 CZY90E 71717497 IC50 = 25 nM T12119 CW5FD9 71717498 IC50 = 25 nM T12119 C3GDC4 71717499 IC50 = 27 nM T12119 CH86VC 71717500 IC50 = 19 nM T12119 CV74QE 71717501 IC50 = 20 nM T12119 COE25L 71717502 IC50 = 21 nM T12119 CG0AK5 71717503 IC50 = 22 nM T12119 C2TN3U 71717504 IC50 = 22 nM T12119 C7HA3R 71717507 IC50 = 34001.65 nM T12119 CQK3J1 71717508 IC50 = 17 nM T12119 CLX7P9 71717509 IC50 = 11 nM T12119 C1YJU6 71717511 IC50 = 37350.81 nM T12119 C60LCK 71717512 IC50 = 25698.04 nM T12119 CZKG01 71717513 IC50 = 10000 nM T12119 C0FX1V 71717514 IC50 = 12459.48 nM T12119 CCE8F2 71717515 IC50 = 12 nM T12119 C5P8IS 71717516 IC50 = 12 nM T12119 CN78EX 71717517 IC50 = 8 nM T12119 CCIB47 71717518 IC50 = 8.4 nM T12119 CXWC82 71717519 IC50 = 3.6 nM T12119 C70EQX 71717520 IC50 = 4.1 nM T12119 CCKY69 71717526 IC50 = 8600.03 nM T12119 CH5CE0 71717527 IC50 = 8999.12 nM T12119 C4QN5I 71717528 IC50 = 10000 nM T12119 C9KV4B 71717529 IC50 = 10000 nM T12119 CQS0P4 71717530 IC50 = 3860.11 nM T12119 CGZ2K7 71717531 IC50 = 4160.06 nM T12119 C76NIM 71717532 IC50 = 4269.73 nM T12119 CO09AY 71717533 IC50 = 4300.31 nM T12119 CMYG42 71717534 IC50 = 6299.41 nM T12119 CUB6X8 71717535 IC50 = 6440.21 nM T12119 CI0ZB4 71717536 IC50 = 2.3 nM T12119 C2OP0D 71717537 IC50 = 2.7 nM T12119 CW8K4Q 71717538 IC50 = 2.7 nM T12119 CC4W1Y 71717539 IC50 = 0.7 nM T12119 CC7HK5 71717540 IC50 = 0.7 nM T12119 CQ4IV7 71717541 IC50 = 3170.3 nM T12119 CG53VX 71717542 IC50 = 3400.17 nM T12119 CNX7F2 71717543 IC50 = 2700.23 nM T12119 C3SD2U 71717544 IC50 = 2800.27 nM T12119 C3UTP4 71717545 IC50 = 2900.01 nM T12119 CXFA25 71717546 IC50 = 2900.01 nM T12119 C5HQ3I 71717547 IC50 = 2999.85 nM T12119 CHAL16 71717548 IC50 = 2189.78 nM T12119 CJXV13 71717549 IC50 = 2199.89 nM T12119 CM9SL4 71717550 IC50 = 2199.89 nM T12119 CQ3GS5 71717551 IC50 = 2279.82 nM T12119 CV9U2H 71717552 IC50 = 2380.13 nM T12119 C0SB9G 71717553 IC50 = 2399.94 nM T12119 C2LD9U 71717554 IC50 = 2399.94 nM T12119 C7R3LI 71717555 IC50 = 2499.77 nM T12119 C4JEG8 71717556 IC50 = 1900.2 nM T12119 C3BZX2 71717557 IC50 = 1980.16 nM T12119 CT62SI 71717560 IC50 = 2030.02 nM T12119 CBMY78 71717561 IC50 = 2030.02 nM T12119 C37LIE 71717562 IC50 = 2050.22 nM T12119 CM4LI9 71717563 IC50 = 1299.87 nM T12119 CX43JE 71717564 IC50 = 1320.08 nM T12119 C6G8NY 71717565 IC50 = 1389.95 nM T12119 CMY01O 71717566 IC50 = 1599.93 nM T12119 C5AH8O 71717567 IC50 = 1699.81 nM T12119 C70MWE 71717568 IC50 = 1000 nM T12119 CD5JP3 71717569 IC50 = 1000 nM T12119 C8QTR2 71717572 IC50 = 1079.94 nM T12119 C5ONB1 71717573 IC50 = 1100.02 nM T12119 C34WZJ 71717574 IC50 = 1130.06 nM T12119 C4MWA5 71717575 IC50 = 1200.05 nM T12119 CWGM51 71717576 IC50 = 1000 nM T12119 CS8YA5 71717991 IC50 = 989.92 nM T12119 CBT2R9 71717992 IC50 = 1000 nM T12119 CHU8A9 71717993 IC50 = 1000 nM T12119 C8RKN7 71717994 IC50 = 739.95 nM T12119 C7W5XG 71717995 IC50 = 770.02 nM T12119 CO7IN3 71717996 IC50 = 840.04 nM T12119 CPG38I 71717997 IC50 = 840.04 nM T12119 COK4T8 71718004 IC50 = 560.02 nM T12119 C9Y0XW 71718005 IC50 = 570.03 nM T12119 CX65MG 71718006 IC50 = 679.99 nM T12119 CZ94IL 71718007 IC50 = 729.96 nM T12119 CSK39X 71718008 IC50 = 479.95 nM T12119 CQ05HL 71718009 IC50 = 479.95 nM T12119 C17ZMY 71718010 IC50 = 490 nM T12119 CNCW13 71718011 IC50 = 500.03 nM T12119 CVI86J 71718016 IC50 = 540.01 nM T12119 CEQ1Y0 71718017 IC50 = 340.02 nM T12119 CG8V3O 71718018 IC50 = 350.03 nM T12119 C2B1LZ 71718019 IC50 = 390.03 nM T12119 CF1N3V 71718020 IC50 = 299.99 nM T12119 C5PH2Q 71718025 IC50 = 310.03 nM T12119 C7W2ZU 71718026 IC50 = 219.99 nM T12119 CIW05Y 71718027 IC50 = 229.99 nM T12119 CS56QP 71718028 IC50 = 229.99 nM T12119 CW5TL7 71718029 IC50 = 229.99 nM T12119 CLV0H1 71718030 IC50 = 239.99 nM T12119 C0CY2Z 71718031 IC50 = 249.98 nM T12119 CJA3L8 71718032 IC50 = 260.02 nM T12119 C5V4AI 71718033 IC50 = 260.02 nM T12119 CKT4N1 71718038 IC50 = 169.98 nM T12119 C6WY2C 71718039 IC50 = 190.02 nM T12119 CV8MR4 71718040 IC50 = 199.99 nM T12119 C9CZ4Y 71718041 IC50 = 129.99 nM T12119 C3AP7Q 71718042 IC50 = 139.99 nM T12119 C9NE2I 71718043 IC50 = 139.99 nM T12119 CR3Z1C 71718044 IC50 = 150 nM T12119 CVGT29 71718055 IC50 = 100 nM T12119 CM4H1Y 71718056 IC50 = 100 nM T12119 CBUO30 71718057 IC50 = 110 nM T12119 C61OCQ 71718058 IC50 = 110 nM T12119 C9A1VJ 71718059 IC50 = 110 nM T12119 C7FN3J 71718060 IC50 = 120.01 nM T12119 C5OHL0 71718061 IC50 = 81 nM T12119 CLSB75 71718062 IC50 = 88 nM T12119 CWD7Z0 71718068 IC50 = 96.01 nM T12119 CEVJ08 71718069 IC50 = 60.01 nM T12119 C0FDB6 71718070 IC50 = 65.99 nM T12119 CN8X2S 71718071 IC50 = 67 nM T12119 C0TK9Q 71718072 IC50 = 28 nM T12119 CXQ6Z4 71718073 IC50 = 70 nM T12119 CJUA26 71718074 IC50 = 71.01 nM T12119 CJ0FI9 71718075 IC50 = 71.99 nM T12119 C8KMT5 71718076 IC50 = 75.01 nM T12119 CDR1K9 71718077 IC50 = 40 nM T12119 C0MTX4 71718078 IC50 = 45 nM T12119 CTV86D 71718086 IC50 = 50 nM T12119 C3Z7EK 71718087 IC50 = 56 nM T12119 CY8IK7 71718088 IC50 = 31 nM T12119 CUH73G 71718089 IC50 = 36 nM T12119 CEM7I3 71718090 IC50 = 23 nM T12119 C6E8ZA 71718091 IC50 = 23 nM T12119 CBV2T7 71718092 IC50 = 25 nM T12119 CH3L0R 71718093 IC50 = 25 nM T12119 CKB07T 71718097 IC50 = 28 nM T12119 C8SL2X 71718098 IC50 = 30 nM T12119 C6L4NF 71718099 IC50 = 30 nM T12119 CB60ZY 71718100 IC50 = 20 nM T12119 C6ZJ7S 71718101 IC50 = 21 nM T12119 C3EJ7I 71718102 IC50 = 22 nM T12119 CVL25J 71718104 IC50 = 32991.34 nM T12119 CHK16A 71718105 IC50 = 35917 nM T12119 CV7TG2 71718106 IC50 = 36846.82 nM T12119 CD23CV 71718107 IC50 = 15 nM T12119 CRFJ80 71718108 IC50 = 15 nM T12119 C3DNM7 71718109 IC50 = 15 nM T12119 C3BAQ6 71718110 IC50 = 10 nM T12119 CX0UQ3 71718111 IC50 = 11 nM T12119 C56XLB 71718112 IC50 = 11 nM T12119 C5CHA2 71718113 IC50 = 11 nM T12119 CL5P9F 71718115 IC50 = 15000.3 nM T12119 C30KIV 71718116 IC50 = 18001.14 nM T12119 C6TN5R 71718117 IC50 = 18001.14 nM T12119 CJOV96 71718118 IC50 = 21702.01 nM T12119 C8DUW6 71718119 IC50 = 22961.49 nM T12119 C87FZU 71718120 IC50 = 23431.5 nM T12119 CO3HC4 71718121 IC50 = 10000 nM T12119 C3QBT9 71718122 IC50 = 10000 nM T12119 C2SKQ6 71718123 IC50 = 10000 nM T12119 CE5DB9 71718124 IC50 = 5.901 nM T12119 CAF91S 71718125 IC50 = 6.4 nM T12119 C5C9NF 71718126 IC50 = 7 nM T12119 C89GSF 71718127 IC50 = 7 nM T12119 C7ID6W 71718128 IC50 = 8.4 nM T12119 C0EVI7 71718129 IC50 = 4.8 nM T12119 C56DFL 71718138 IC50 = 12708.67 nM T12119 CRH4X8 71718139 IC50 = 12858.79 nM T12119 CYI26Z 71718140 IC50 = 3980.16 nM T12119 CT6IQ5 71718141 IC50 = 4799.54 nM T12119 CWA8S9 71718142 IC50 = 4900.04 nM T12119 CAS9F8 71718143 IC50 = 5679.37 nM T12119 C9A7SR 71718144 IC50 = 6200.12 nM T12119 CIGU69 71718145 IC50 = 1.5 nM T12119 CBJD61 71718146 IC50 = 2.4 nM T12119 CT2Z4C 71718147 IC50 = 1.4 nM T12119 CA5YO9 71718148 IC50 = 7479.97 nM T12119 C0S7NV 71718149 IC50 = 3080.35 nM T12119 CN27HU 71718150 IC50 = 3299.89 nM T12119 CWJY35 71718151 IC50 = 3489.8 nM T12119 C8N0FX 71718152 IC50 = 2600.16 nM T12119 C8D7MI 71718153 IC50 = 2949.85 nM T12119 C37UHX 71718157 IC50 = 2999.85 nM T12119 CGC25D 71718158 IC50 = 2999.85 nM T12119 CMTJ56 71718159 IC50 = 2999.85 nM T12119 CNXZ89 71718160 IC50 = 2199.89 nM T12119 C3MRK8 71718161 IC50 = 2350.17 nM T12119 CP93XC 71718162 IC50 = 1729.82 nM T12119 CFW10L 71718163 IC50 = 1800.11 nM T12119 C41HRS 71718164 IC50 = 1850.12 nM T12119 CA0R5Q 71718171 IC50 = 1999.86 nM T12119 CR3F8L 71718172 IC50 = 1299.87 nM T12119 CCTV92 71718173 IC50 = 1299.87 nM T12119 CPK1G7 71718174 IC50 = 1299.87 nM T12119 CHM5K9 71718175 IC50 = 1580.16 nM T12119 CC0EQ5 71718176 IC50 = 1599.93 nM T12119 CCX3H0 71718177 IC50 = 1699.81 nM T12119 C4SWF3 71718187 IC50 = 1200.05 nM T12119 CD0ZI9 71718188 IC50 = 1290.03 nM T12119 CIVS51 71718189 IC50 = 1000 nM T12119 C9QN5H 71718190 IC50 = 1000 nM T12119 CTNM52 71718191 IC50 = 1000 nM T12119 CSZ16M 71718192 IC50 = 1000 nM T12119 C63IWN 71718193 IC50 = 1000 nM T12119 CJ1SA9 71718605 IC50 = 939.94 nM T12119 C2RDM0 71718606 IC50 = 970.06 nM T12119 C68CTU 71718607 IC50 = 989.92 nM T12119 CI6P0S 71718608 IC50 = 1000 nM T12119 COG60R 71718609 IC50 = 1000 nM T12119 CUW48S 71718610 IC50 = 1000 nM T12119 C0I1DY 71718611 IC50 = 1000 nM T12119 CQK42W 71718612 IC50 = 759.98 nM T12119 C3VOJ1 71718613 IC50 = 770.02 nM T12119 CQ78CJ 71718614 IC50 = 810.03 nM T12119 CNA4J6 71718615 IC50 = 819.97 nM T12119 C75XBN 71718616 IC50 = 819.97 nM T12119 C69VQW 71718617 IC50 = 849.96 nM T12119 C57UHB 71718623 IC50 = 659.93 nM T12119 C6QX8N 71718624 IC50 = 689.92 nM T12119 C2XF6K 71718625 IC50 = 700 nM T12119 C30LVS 71718626 IC50 = 710.07 nM T12119 C0O7TI 71718627 IC50 = 729.96 nM T12119 C78NSZ 71718628 IC50 = 449.99 nM T12119 CG0BV9 71718629 IC50 = 470 nM T12119 C7TM8H 71718630 IC50 = 465 nM T12119 COM9W1 71718631 IC50 = 479.95 nM T12119 CWAR24 71718632 IC50 = 500.03 nM T12119 CH3T4J 71718640 IC50 = 530.03 nM T12119 CG5S2K 71718641 IC50 = 360 nM T12119 C6R7HB 71718642 IC50 = 419.95 nM T12119 C8EZU5 71718643 IC50 = 270.02 nM T12119 CN8E3Q 71718644 IC50 = 270.02 nM T12119 C3A5TJ 71718652 IC50 = 219.99 nM T12119 CY1DR8 71718653 IC50 = 260.02 nM T12119 CU2L9A 71718654 IC50 = 169.98 nM T12119 C0BJ2O 71718660 IC50 = 209.99 nM T12119 C1L7OZ 71718661 IC50 = 209.99 nM T12119 C6L2NB 71718662 IC50 = 129.99 nM T12119 C5ZMD9 71718663 IC50 = 129.99 nM T12119 CVOJ63 71718664 IC50 = 139.99 nM T12119 CW1BD6 71718665 IC50 = 139.99 nM T12119 CGX6Y9 71718666 IC50 = 139.99 nM T12119 CH91CA 71718667 IC50 = 139.99 nM T12119 C18XQA 71718673 IC50 = 159.99 nM T12119 C7APJ0 71718674 IC50 = 110 nM T12119 C5I0BF 71718675 IC50 = 88 nM T12119 CY3PG6 71718680 IC50 = 89.99 nM T12119 C7SY1A 71718681 IC50 = 60.01 nM T12119 C74TZY 71718682 IC50 = 70 nM T12119 C13TGI 71718683 IC50 = 48 nM T12119 CLE3H9 71718687 IC50 = 90 nM T12119 CF3J2U 71718688 IC50 = 53 nM T12119 C24BJI 71718689 IC50 = 56 nM T12119 CZA4E3 71718690 IC50 = 31 nM T12119 C2TM5B 71718691 IC50 = 34 nM T12119 CG56DC 71718692 IC50 = 35 nM T12119 CVY46H 71718693 IC50 = 39 nM T12119 C2WK4I 71718697 IC50 = 26 nM T12119 CR3DO8 71718698 IC50 = 30 nM T12119 CD90KU 71718699 IC50 = 20 nM T12119 C6NA1C 71718700 IC50 = 20 nM T12119 C0O8EZ 71718701 IC50 = 21 nM T12119 C45BNQ 71718702 IC50 = 22 nM T12119 C8QW5U 71718703 IC50 = 29998.53 nM T12119 CPM16K 71718704 IC50 = 31002.73 nM T12119 C82ECS 71718705 IC50 = 35999.79 nM T12119 CIK6B5 71718706 IC50 = 35999.79 nM T12119 CN67WH 71718707 IC50 = 14 nM T12119 C50LGE 71718708 IC50 = 14 nM T12119 C9VZG2 71718709 IC50 = 17 nM T12119 C3Z7HP 71718710 IC50 = 17 nM T12119 CT34AP 71718711 IC50 = 9.899 nM T12119 CKW47U 71718712 IC50 = 10 nM T12119 CF9HD1 71718713 IC50 = 11 nM T12119 CUI3T6 71718715 IC50 = 13999.1 nM T12119 C3XU9H 71718716 IC50 = 15000.3 nM T12119 CZ39LN 71718717 IC50 = 15409.91 nM T12119 CO9CH5 71718718 IC50 = 10000 nM T12119 CVDZ25 71718719 IC50 = 11000.19 nM T12119 CN7Z9H 71718720 IC50 = 11000.19 nM T12119 C0IPV3 71718721 IC50 = 12119.93 nM T12119 C1DKH4 71718722 IC50 = 11 nM T12119 C1FBJ5 71718723 IC50 = 7.399 nM T12119 C9CR3E 71718724 IC50 = 4.2 nM T12119 CGZ01J 71718725 IC50 = 4.2 nM T12119 CW38FM 71718726 IC50 = 4.8 nM T12119 CW4I3T 71718731 IC50 = 12511.23 nM T12119 C9ZE3P 71718732 IC50 = 8699.61 nM T12119 C2EZ7F 71718733 IC50 = 10000 nM T12119 C9D1ML 71718734 IC50 = 10000 nM T12119 C7DL3J 71718735 IC50 = 3900.32 nM T12119 C8Z2CV 71718736 IC50 = 6899.22 nM T12119 CBC2U5 71718737 IC50 = 1.7 nM T12119 C6TWV7 71718738 IC50 = 2.1 nM T12119 C8AL2K 71718739 IC50 = 2.3 nM T12119 CQ6IC5 71718740 IC50 = 2.4 nM T12119 C6MLD8 71718741 IC50 = 0.8999 nM T12119 C5KL7V 71718742 IC50 = 3299.89 nM T12119 CWHP07 71718743 IC50 = 3400.17 nM T12119 C9XO7H 71718744 IC50 = 3410.36 nM T12119 C5FMR8 71718745 IC50 = 3539.97 nM T12119 CUB3R6 71718746 IC50 = 3599.98 nM T12119 C49TJB 71718747 IC50 = 2600.16 nM T12119 C9JXS2 71718748 IC50 = 2600.16 nM T12119 CIB63K 71718749 IC50 = 2900.01 nM T12119 CTJ3H8 71718750 IC50 = 2979.89 nM T12119 C43KGM 71718751 IC50 = 2999.85 nM T12119 CVS1F9 71718755 IC50 = 2999.85 nM T12119 CB97VR 71718756 IC50 = 2170.2 nM T12119 CC3LV1 71718757 IC50 = 2210.04 nM T12119 CEW76D 71718758 IC50 = 2250.09 nM T12119 CEI0J1 71718759 IC50 = 2299.85 nM T12119 CEZ8S4 71718760 IC50 = 2499.77 nM T12119 CHM84A 71718761 IC50 = 2499.77 nM T12119 CDF1K6 71718762 IC50 = 2499.77 nM T12119 CA1N0L 71718763 IC50 = 2529.88 nM T12119 CR98MO 71718764 IC50 = 2590 nM T12119 CN7J1A 71718765 IC50 = 1800.11 nM T12119 CN60MA 71718766 IC50 = 1800.11 nM T12119 CTAM64 71718767 IC50 = 1810.09 nM T12119 CO8AG2 71718772 IC50 = 1999.86 nM T12119 CJ41XS 71718773 IC50 = 2099.91 nM T12119 CD1Z6T 71718774 IC50 = 2099.91 nM T12119 CE67NZ 71718775 IC50 = 1599.93 nM T12119 CMH2P6 71718780 IC50 = 1039.92 nM T12119 CKD83W 71718781 IC50 = 1100.02 nM T12119 CA91TN 71718782 IC50 = 1100.02 nM T12119 CF8J2H 71718783 IC50 = 1200.05 nM T12119 CZW71H 71718784 IC50 = 1000 nM T12119 C0T2HE 71718785 IC50 = 1000 nM T12119 CNA45C 71718786 IC50 = 1000 nM T12119 C6ZG1V 71719221 IC50 = 1000 nM T12119 C4K9TC 71719222 IC50 = 1000 nM T12119 CN1MT7 71719223 IC50 = 739.95 nM T12119 C6TNR0 71719229 IC50 = 550.05 nM T12119 CF6Q0L 71719230 IC50 = 579.96 nM T12119 CC2M3J 71719231 IC50 = 579.96 nM T12119 CK78TN 71719232 IC50 = 590.07 nM T12119 C7E0JC 71719233 IC50 = 629.94 nM T12119 C4F7QT 71719234 IC50 = 430.03 nM T12119 CS6I0V 71719235 IC50 = 449.99 nM T12119 CJ70AT 71719236 IC50 = 490 nM T12119 CU4VD9 71719237 IC50 = 510.04 nM T12119 C8K2QE 71719242 IC50 = 540.01 nM T12119 CT8UC9 71719243 IC50 = 340.02 nM T12119 C78DIM 71719244 IC50 = 350.03 nM T12119 CC2F1S 71719245 IC50 = 370 nM T12119 C4OHU0 71719246 IC50 = 390.03 nM T12119 C1YW9Q 71719247 IC50 = 400.04 nM T12119 C7YW0V 71719248 IC50 = 410.02 nM T12119 CY3PU1 71719249 IC50 = 430.03 nM T12119 CN7IQ4 71719250 IC50 = 430.03 nM T12119 CX5OL0 71719251 IC50 = 299.99 nM T12119 C5A8PR 71719258 IC50 = 299.99 nM T12119 C7C5JM 71719259 IC50 = 310.03 nM T12119 CPE62B 71719260 IC50 = 219.99 nM T12119 C6HQE1 71719261 IC50 = 229.99 nM T12119 CH79XU 71719262 IC50 = 260.02 nM T12119 CTI42W 71719267 IC50 = 169.98 nM T12119 CAN7J0 71719268 IC50 = 180.01 nM T12119 C9GUE7 71719269 IC50 = 190.02 nM T12119 CHNC09 71719270 IC50 = 190.02 nM T12119 CAG06O 71719271 IC50 = 190.02 nM T12119 CG7DY0 71719272 IC50 = 190.02 nM T12119 C2CJV3 71719273 IC50 = 209.99 nM T12119 CBXP76 71719274 IC50 = 129.99 nM T12119 C31KAO 71719275 IC50 = 139.99 nM T12119 C9IO4W 71719276 IC50 = 159.99 nM T12119 C87GCK 71719282 IC50 = 159.99 nM T12119 C95DVU 71719283 IC50 = 110 nM T12119 CHVW71 71719284 IC50 = 120.01 nM T12119 CZ7O3P 71719285 IC50 = 120.01 nM T12119 CJH5S7 71719286 IC50 = 120.01 nM T12119 C93TNY 71719287 IC50 = 120.01 nM T12119 C8Z1DP 71719288 IC50 = 80 nM T12119 C6I3UV 71719289 IC50 = 80 nM T12119 C69YPD 71719290 IC50 = 81 nM T12119 CDX65G 71719291 IC50 = 88 nM T12119 CPQ2D0 71719294 IC50 = 90.99 nM T12119 CTB2Y6 71719295 IC50 = 96.01 nM T12119 C3F6SE 71719296 IC50 = 97.01 nM T12119 CAUC02 71719297 IC50 = 57 nM T12119 CBSQ38 71719298 IC50 = 65.99 nM T12119 CZ1SP5 71719299 IC50 = 75.01 nM T12119 CK6AG9 71719300 IC50 = 77 nM T12119 CQ9AF0 71719301 IC50 = 77 nM T12119 CSA57C 71719302 IC50 = 40 nM T12119 CZ41VW 71719303 IC50 = 44 nM T12119 C21GEV 71719304 IC50 = 46 nM T12119 CYL79O 71719309 IC50 = 53 nM T12119 C3I0OF 71719310 IC50 = 33 nM T12119 CK3TW4 71719311 IC50 = 34 nM T12119 CP0CD5 71719312 IC50 = 35 nM T12119 CBTY30 71719313 IC50 = 39 nM T12119 CG2U4E 71719314 IC50 = 22 nM T12119 C3WFI8 71719315 IC50 = 27 nM T12119 CW67VK 71719316 IC50 = 29 nM T12119 CN3FD7 71719317 IC50 = 19 nM T12119 CTR3S9 71719318 IC50 = 12 nM T12119 C2DKO8 71719319 IC50 = 12 nM T12119 C2A9NY 71719320 IC50 = 12 nM T12119 C2F0IS 71719323 IC50 = 33736.5 nM T12119 CS2D7O 71719324 IC50 = 36082.78 nM T12119 CU5EQ9 71719325 IC50 = 17 nM T12119 CW4PE3 71719326 IC50 = 9.399 nM T12119 CGOS70 71719327 IC50 = 11 nM T12119 CZ8D3R 71719328 IC50 = 11 nM T12119 C04HZJ 71719329 IC50 = 51003.5 nM T12119 C72RVE 71719330 IC50 = 15059.13 nM T12119 CX4A7O 71719331 IC50 = 25491.77 nM T12119 CHIG08 71719332 IC50 = 10000 nM T12119 CLTD46 71719333 IC50 = 5.1 nM T12119 C0F3GW 71719334 IC50 = 7.8 nM T12119 C5RAQ1 71719335 IC50 = 4.6 nM T12119 C7O0HI 71719336 IC50 = 4.7 nM T12119 C2YTE5 71719344 IC50 = 8869.52 nM T12119 C6THB0 71719345 IC50 = 9189.67 nM T12119 CVL2A9 71719346 IC50 = 9899.2 nM T12119 C4GLF9 71719347 IC50 = 10000 nM T12119 CQO7Z6 71719348 IC50 = 3900.32 nM T12119 C0T1CH 71719349 IC50 = 4.8 nM T12119 CPL34E 71719350 IC50 = 2.5 nM T12119 C2LYA9 71719351 IC50 = 2.5 nM T12119 CJZ0V1 71719352 IC50 = 3059.85 nM T12119 C2S8YQ 71719353 IC50 = 3110.28 nM T12119 CNFC71 71719354 IC50 = 3299.89 nM T12119 CUY51I 71719355 IC50 = 3400.17 nM T12119 C16XUQ 71719356 IC50 = 3400.17 nM T12119 C9AY0W 71719357 IC50 = 3500.26 nM T12119 CWL3S4 71719358 IC50 = 3760.11 nM T12119 CXJ56Q 71719359 IC50 = 3800.14 nM T12119 CFG7A9 71719360 IC50 = 2600.16 nM T12119 CFXT35 71719361 IC50 = 2700.23 nM T12119 CL4WP9 71719362 IC50 = 2779.71 nM T12119 CGHY01 71719363 IC50 = 2800.27 nM T12119 C7NL8Q 71719364 IC50 = 2409.91 nM T12119 CAE8I9 71719365 IC50 = 2499.77 nM T12119 C83YCE 71719366 IC50 = 1790.19 nM T12119 C6H1RX 71719367 IC50 = 1810.09 nM T12119 CAS4I3 71719368 IC50 = 1869.82 nM T12119 C7QUW1 71719369 IC50 = 1900.2 nM T12119 CIH5U8 71719371 IC50 = 2089.78 nM T12119 C2YGZ7 71719372 IC50 = 1369.94 nM T12119 C50YNW 71719373 IC50 = 1429.88 nM T12119 CO51XI 71719374 IC50 = 1469.94 nM T12119 C86PUZ 71719375 IC50 = 1500.03 nM T12119 CU6PH0 71719376 IC50 = 1570 nM T12119 CKZ3S4 71719381 IC50 = 1119.95 nM T12119 CLT0N4 71719382 IC50 = 1189.87 nM T12119 C50ZGW 71719383 IC50 = 1200.05 nM T12119 C2EL0X 71719384 IC50 = 1299.87 nM T12119 CA5QH4 71719385 IC50 = 1000 nM T12119 CGC58T 71719386 IC50 = 1000 nM T12119 CB98LN 71719387 IC50 = 1000 nM T12119 CZI12Y 71719388 IC50 = 1000 nM T12119 CW2LY6 71719389 IC50 = 1000 nM T12119 C5GBQ7 71719390 IC50 = 920.03 nM T12119 C7Z4ED 71719831 IC50 = 949.95 nM T12119 COTI35 71719832 IC50 = 1000 nM T12119 CP3ZT4 71719833 IC50 = 810.03 nM T12119 CK6Q9B 71719834 IC50 = 899.91 nM T12119 CQEX07 71719839 IC50 = 739.95 nM T12119 C14JHN 71719840 IC50 = 449.99 nM T12119 C0JPN1 71719841 IC50 = 470 nM T12119 CAJ5V7 71719845 IC50 = 540.01 nM T12119 CC5N8P 71719846 IC50 = 350.03 nM T12119 CQ76XJ 71719847 IC50 = 350.03 nM T12119 CAR98W 71719848 IC50 = 360 nM T12119 CZK23L 71719849 IC50 = 360 nM T12119 CWP14U 71719850 IC50 = 390.03 nM T12119 CRVM70 71719851 IC50 = 260.02 nM T12119 C2M0AU 71719852 IC50 = 299.99 nM T12119 CANF64 71719853 IC50 = 299.99 nM T12119 C9TGN4 71719860 IC50 = 299.99 nM T12119 CDIM32 71719861 IC50 = 329.99 nM T12119 CZI86Y 71719862 IC50 = 229.99 nM T12119 C5T7UG 71719863 IC50 = 239.99 nM T12119 CJ2SC6 71719864 IC50 = 239.99 nM T12119 CMI75O 71719868 IC50 = 199.99 nM T12119 CRKB05 71719869 IC50 = 159.99 nM T12119 C5ZMS0 71719870 IC50 = 159.99 nM T12119 CHXG64 71719875 IC50 = 100 nM T12119 CA2CH1 71719876 IC50 = 110 nM T12119 C0REO9 71719877 IC50 = 120.01 nM T12119 CY4RJ9 71719878 IC50 = 120.01 nM T12119 C9VH2T 71719879 IC50 = 120.01 nM T12119 CAO68K 71719880 IC50 = 79 nM T12119 C6XO0Q 71719881 IC50 = 80 nM T12119 C04BFW 71719882 IC50 = 83 nM T12119 CDLF98 71719883 IC50 = 87 nM T12119 CE0T1K 71719887 IC50 = 89.99 nM T12119 CPES10 71719888 IC50 = 70 nM T12119 C4O8JN 71719889 IC50 = 45 nM T12119 C58JVO 71719899 IC50 = 30 nM T12119 CB9VJ8 71719900 IC50 = 31 nM T12119 CSOL35 71719901 IC50 = 32 nM T12119 CX85EL 71719902 IC50 = 34 nM T12119 CY6D2J 71719903 IC50 = 34 nM T12119 C5HT0S 71719904 IC50 = 40 nM T12119 CL0O5N 71719912 IC50 = 30 nM T12119 CJ31QS 71719913 IC50 = 19 nM T12119 CYQH30 71719914 IC50 = 20 nM T12119 CA42SN 71719915 IC50 = 20 nM T12119 CN8YC4 71719916 IC50 = 22 nM T12119 C1PM2H 71719917 IC50 = 22 nM T12119 CXBF28 71719918 IC50 = 13 nM T12119 C4ELW8 71719919 IC50 = 29998.53 nM T12119 C6FJW0 71719920 IC50 = 30902.95 nM T12119 C0AXF2 71719921 IC50 = 14 nM T12119 C8TY7U 71719922 IC50 = 17 nM T12119 C30WQM 71719923 IC50 = 17 nM T12119 C82INW 71719924 IC50 = 9.601 nM T12119 CN6W1U 71719925 IC50 = 10 nM T12119 C5Z7RX 71719926 IC50 = 11 nM T12119 C5UW8R 71719929 IC50 = 38707.93 nM T12119 COB5H2 71719930 IC50 = 16210.63 nM T12119 C0WLZ2 71719931 IC50 = 18450.15 nM T12119 C7GPC0 71719932 IC50 = 24468.09 nM T12119 CDU9C4 71719933 IC50 = 10000 nM T12119 C56COE 71719934 IC50 = 10000 nM T12119 CVO12U 71719935 IC50 = 11590.44 nM T12119 C7XRA9 71719936 IC50 = 12000.52 nM T12119 CIT4P9 71719937 IC50 = 12000.52 nM T12119 C5XEH8 71719938 IC50 = 12000.52 nM T12119 CDL1U0 71719939 IC50 = 6.299 nM T12119 CMLE56 71719945 IC50 = 9200.26 nM T12119 C1ALS5 71719946 IC50 = 10000 nM T12119 C59FXL 71719947 IC50 = 10000 nM T12119 C9T0JC 71719948 IC50 = 4600.45 nM T12119 C1RT0J 71719949 IC50 = 6000.67 nM T12119 C5QX8G 71719950 IC50 = 1.8 nM T12119 CJ6AV3 71719951 IC50 = 2.4 nM T12119 C86OTM 71719952 IC50 = 3.1 nM T12119 C43PIS 71719953 IC50 = 1.1 nM T12119 C4FG1V 71719954 IC50 = 1.4 nM T12119 C2EM5Z 71719955 IC50 = 7100.68 nM T12119 C35IDS 71719956 IC50 = 3100.27 nM T12119 CZI28H 71719957 IC50 = 3139.79 nM T12119 CBL7W2 71719958 IC50 = 3139.79 nM T12119 CES07K 71719959 IC50 = 3379.87 nM T12119 C1ELK9 71719960 IC50 = 3400.17 nM T12119 CZCF53 71719962 IC50 = 2999.85 nM T12119 CLKU73 71719963 IC50 = 2299.85 nM T12119 C0YVS1 71719964 IC50 = 2299.85 nM T12119 CFI01B 71719965 IC50 = 2450.19 nM T12119 C46RTQ 71719966 IC50 = 1900.2 nM T12119 CY74OL 71719968 IC50 = 1999.86 nM T12119 CYKH61 71719969 IC50 = 1440.12 nM T12119 C1AU0O 71719970 IC50 = 1599.93 nM T12119 CJ1VP9 71719971 IC50 = 1599.93 nM T12119 CF9Z7S 71719972 IC50 = 1599.93 nM T12119 CDC0M6 71719980 IC50 = 1050.03 nM T12119 C5U9KC 71719981 IC50 = 1100.02 nM T12119 CW21DS 71719982 IC50 = 1200.05 nM T12119 CE78NX 71719983 IC50 = 1000 nM T12119 CM1Z6X 71719984 IC50 = 1000 nM T12119 C0ZS1M 71719985 IC50 = 1000 nM T12119 CYJ82M 71719986 IC50 = 1000 nM T12119 C1M5UG 71719987 IC50 = 1000 nM T12119 CAGP03 71719988 IC50 = 1000 nM T12119 C2ED6S 71719989 IC50 = 1000 nM T12119 C26BPR 71720438 IC50 = 1000 nM T12119 CQ4NF3 71720439 IC50 = 1000 nM T12119 C6WB8G 71720440 IC50 = 780.01 nM T12119 C0P9ED 71720441 IC50 = 819.97 nM T12119 C4JRG8 71720448 IC50 = 579.96 nM T12119 CW85DP 71720449 IC50 = 629.94 nM T12119 C03TDX 71720450 IC50 = 719.95 nM T12119 C2Z5LE 71720451 IC50 = 719.95 nM T12119 C7K9MR 71720452 IC50 = 739.95 nM T12119 C6E5YB 71720453 IC50 = 510.04 nM T12119 CSX08O 71720459 IC50 = 540.01 nM T12119 CUN9B6 71720460 IC50 = 340.02 nM T12119 CY4AH2 71720461 IC50 = 400.04 nM T12119 CD1LC3 71720462 IC50 = 410.02 nM T12119 C6G5SI 71720463 IC50 = 430.03 nM T12119 CD6SL0 71720469 IC50 = 299.99 nM T12119 CMDI34 71720470 IC50 = 319.96 nM T12119 C7BL3K 71720471 IC50 = 329.99 nM T12119 CR70IZ 71720472 IC50 = 229.99 nM T12119 C8YA4W 71720473 IC50 = 229.99 nM T12119 CKMV37 71720474 IC50 = 239.99 nM T12119 CV9QM8 71720475 IC50 = 239.99 nM T12119 C4B8CZ 71720480 IC50 = 169.98 nM T12119 CR7S3B 71720481 IC50 = 180.01 nM T12119 CPH7V4 71720482 IC50 = 190.02 nM T12119 CKJ95I 71720483 IC50 = 190.02 nM T12119 CN8V0O 71720484 IC50 = 120.01 nM T12119 CX4M1C 71720485 IC50 = 139.99 nM T12119 CJS50E 71720486 IC50 = 159.99 nM T12119 C86XHB 71720497 IC50 = 159.99 nM T12119 C1QC4N 71720498 IC50 = 100 nM T12119 CMJ1K4 71720499 IC50 = 110 nM T12119 C3DCB1 71720508 IC50 = 97.01 nM T12119 CWJN65 71720509 IC50 = 100 nM T12119 CVN2Q1 71720510 IC50 = 57 nM T12119 CXRB98 71720511 IC50 = 62.99 nM T12119 CO3RB1 71720512 IC50 = 64 nM T12119 CEWQ56 71720513 IC50 = 76 nM T12119 CU07OA 71720514 IC50 = 77 nM T12119 C2AKC8 71720515 IC50 = 78 nM T12119 CDGQ30 71720522 IC50 = 50 nM T12119 CS8TX9 71720523 IC50 = 33 nM T12119 C24GTR 71720524 IC50 = 24 nM T12119 CV2WH8 71720528 IC50 = 30 nM T12119 C18BSG 71720529 IC50 = 30 nM T12119 CSCR71 71720530 IC50 = 19 nM T12119 COV3G7 71720531 IC50 = 20 nM T12119 C6U3BT 71720532 IC50 = 22 nM T12119 C5A0GB 71720533 IC50 = 12 nM T12119 C52HXL 71720537 IC50 = 29998.53 nM T12119 C02BXS 71720538 IC50 = 14 nM T12119 CCL36M 71720539 IC50 = 14 nM T12119 CUEO39 71720540 IC50 = 14 nM T12119 C3XHB4 71720541 IC50 = 15 nM T12119 C3IB2G 71720542 IC50 = 16 nM T12119 C7B8UH 71720543 IC50 = 8.5 nM T12119 C0U6PV 71720544 IC50 = 9.2 nM T12119 CM67TB 71720546 IC50 = 54000.78 nM T12119 CWJ9P4 71720547 IC50 = 15000.3 nM T12119 CK57XY 71720548 IC50 = 15881.81 nM T12119 CXH40F 71720549 IC50 = 16531.03 nM T12119 CEJO28 71720550 IC50 = 19230.92 nM T12119 CS4O2A 71720551 IC50 = 23999.38 nM T12119 C9TV2X 71720552 IC50 = 24997.7 nM T12119 CH5XN0 71720553 IC50 = 29998.53 nM T12119 C0HRB8 71720554 IC50 = 10000 nM T12119 CTYK73 71720555 IC50 = 10000 nM T12119 CW64TL 71720556 IC50 = 11000.19 nM T12119 C5TB0O 71720557 IC50 = 12209.56 nM T12119 CJS34M 71720558 IC50 = 5.1 nM T12119 CHB3U7 71720559 IC50 = 5.2 nM T12119 CZ29BJ 71720560 IC50 = 5.901 nM T12119 CKFQ40 71720561 IC50 = 7 nM T12119 C8UGC3 71720562 IC50 = 4.4 nM T12119 CLF21V 71720573 IC50 = 7710.81 nM T12119 C9AI7O 71720574 IC50 = 9170.65 nM T12119 C6EL2U 71720575 IC50 = 9499.48 nM T12119 C6DE4Y 71720576 IC50 = 10000 nM T12119 C51KVG 71720577 IC50 = 10000 nM T12119 C41MGU 71720578 IC50 = 10000 nM T12119 CG4AM6 71720579 IC50 = 4000.37 nM T12119 CHZG71 71720580 IC50 = 4300.31 nM T12119 CNE4L1 71720581 IC50 = 5400.08 nM T12119 CLW2J7 71720582 IC50 = 5500.47 nM T12119 CP80NE 71720583 IC50 = 0.6001 nM T12119 CG21AH 71720584 IC50 = 7299.62 nM T12119 CK8U2I 71720585 IC50 = 7299.62 nM T12119 C5BPM6 71720586 IC50 = 2999.85 nM T12119 CCH6I5 71720587 IC50 = 3299.89 nM T12119 C40STU 71720588 IC50 = 3299.89 nM T12119 C60VEH 71720589 IC50 = 2660.11 nM T12119 C3ZU5M 71720590 IC50 = 2700.23 nM T12119 CB6GC1 71720591 IC50 = 2700.23 nM T12119 CG1PF7 71720593 IC50 = 2199.89 nM T12119 C4J9CT 71720594 IC50 = 2299.85 nM T12119 CUPO90 71720595 IC50 = 2539.8 nM T12119 CXO6M9 71720596 IC50 = 1800.11 nM T12119 CI0V9K 71720597 IC50 = 1900.2 nM T12119 C37HUZ 71720601 IC50 = 1299.87 nM T12119 C4VBM2 71720602 IC50 = 1299.87 nM T12119 C96HXO 71720603 IC50 = 1500.03 nM T12119 CZ6IM8 71720604 IC50 = 1510.08 nM T12119 CZ96YD 71720605 IC50 = 1599.93 nM T12119 CJ4A8C 71720606 IC50 = 1699.81 nM T12119 C9XS1E 71720607 IC50 = 1000 nM T12119 CJK5U4 71720608 IC50 = 1109.94 nM T12119 CVP3U7 71720609 IC50 = 1109.94 nM T12119 C54ANI 71720610 IC50 = 1200.05 nM T12119 C4FIG3 71720611 IC50 = 1229.99 nM T12119 CJ1SQ3 71720612 IC50 = 1000 nM T12119 C3HKF2 71720613 IC50 = 1000 nM T12119 CGKE92 71720614 IC50 = 920.03 nM T12119 CC84RA 71722102 IC50 = 133 nM T12119 C30IKR 71731528 IC50 = 1150 nM T12119 C41QOI 71770953 IC50 = 770 nM T12119 CZE8K5 72188645 IC50 = 1995.26 nM T12119 CJB37T 72201088 IC50 = 251.19 nM T12119 CYMS42 72545669 IC50 = 4 nM T12119 CB87KJ 72548337 IC50 = 1995.26 nM T12119 CCEX08 72949434 IC50 = 6 nM T12119 CDU3T6 73350512 IC50 = 103 nM T12119 CWT18O 73352021 IC50 = 131 nM T12119 CY1G6S 73352027 IC50 = 117 nM T12119 CMR5B8 73353486 IC50 = 137 nM T12119 CP02HY 73354983 IC50 = 101 nM T12119 CB9H2J 74221064 IC50 = 3026 nM T12119 C4OSC2 74221699 IC50 = 134 nM T12119 C0DXB6 74222318 IC50 = 39 nM T12119 CI59EF 74222826 IC50 = 150 nM T12119 C0FVD8 74222919 IC50 = 535 nM T12119 C7OE1X 76309796 IC50 > 30000 nM T12119 CBH4N7 76309797 IC50 = 20000 nM T12119 C10UTF 76310404 IC50 = 27000 nM T12119 C6T1NV 76310406 IC50 > 30000 nM T12119 CC4BK5 76310408 IC50 > 30000 nM T12119 C8M7RN 76310409 IC50 = 26000 nM T12119 CHFC49 76313502 IC50 > 30000 nM T12119 C1PM7H 76314065 IC50 > 30000 nM T12119 CBK0T8 76314067 IC50 > 30000 nM T12119 C20ILA 76314069 IC50 > 30000 nM T12119 C8OQT1 76314070 IC50 = 19000 nM T12119 CI5P8G 76316660 IC50 = 60 nM T12119 CNM4K0 76317019 IC50 = 29000 nM T12119 C32OSF 76317020 IC50 > 30000 nM T12119 CKG5A9 76317629 IC50 > 30000 nM T12119 CQ7JK4 76317631 IC50 = 28000 nM T12119 C4WR1N 76320377 IC50 = 100 nM T12119 CT2R5J 76320732 IC50 > 30000 nM T12119 CVP8U9 76320733 IC50 = 21000 nM T12119 C2RJW0 76320734 IC50 = 16000 nM T12119 CY8NT4 76321352 IC50 = 29000 nM T12119 CRU30A 76321353 IC50 > 30000 nM T12119 C46MFT 76324385 IC50 = 23000 nM T12119 C4W1NV 76324386 IC50 > 30000 nM T12119 CJF20G 76324950 IC50 > 30000 nM T12119 CP3UI7 76327945 IC50 = 21000 nM T12119 CNY5X1 76328517 IC50 > 30000 nM T12119 CX54MA 76328518 IC50 > 30000 nM T12119 C68INR 76331237 IC50 = 700 nM T12119 CINA95 76331591 IC50 = 20000 nM T12119 CCXK29 76332197 IC50 > 30000 nM T12119 CH4K7Q 76332198 IC50 > 30000 nM T12119 C4WO6Y 76332199 IC50 = 22000 nM T12119 CK47NO 76332200 IC50 > 30000 nM T12119 CANB89 76332201 IC50 = 19000 nM T12119 CO2N7R 76335221 IC50 > 30000 nM T12119 C05RSQ 76335223 IC50 = 23000 nM T12119 C8ND6L 76335224 IC50 = 18000 nM T12119 CUO84S 76335833 IC50 > 30000 nM T12119 C39UOX 86267295 IC50 = 140 nM T12119 CV6P7L 86267492 IC50 = 10 nM T12119 CIW2R3 86267733 IC50 = 6 nM T12119 C0EJ1C 86267935 IC50 = 2 nM T12119 C5Z3SK 86268555 IC50 = 74 nM T12119 CRAJ20 86268763 IC50 = 950 nM T12119 CT6W3C 86270135 IC50 = 160 nM T12119 C15BSO 86270136 IC50 = 3 nM T12119 CZL23E 86271138 IC50 > 30000 nM T12119 CK02ZT 86344136 IC50 = 12 nM T12119 CZU43C 86344330 IC50 = 15 nM T12119 C6D5QL 86344510 IC50 = 26 nM T12119 CM3AE5 86344511 IC50 = 27 nM T12119 C1UZ7Y 86344512 IC50 = 17 nM T12119 CJC7V3 86344877 IC50 = 19 nM T12119 C3SIV1 86345235 IC50 = 10 nM T12119 C7J9FE 86687346 IC50 = 160 nM T12119 C0OTF5 86687356 IC50 = 590 nM T12119 C50EDA 86687482 IC50 = 300 nM T12119 CEQ0C1 86687530 IC50 = 320 nM T12119 CTG76E 86687532 IC50 = 140 nM T12119 CQN21C 86687557 IC50 = 150 nM T12119 CFT89Y 86687602 IC50 = 23 nM T12119 CY8JW3 86687604 IC50 = 65 nM T12119 C7OXV8 86687606 IC50 = 49 nM T12119 C63MCA 86687768 IC50 = 19 nM T12119 CJC29A 89544489 IC50 = 17 nM T12119 COK7U5 89545491 IC50 = 82 nM T12119 CAM65C 89545507 IC50 = 0.9 nM T12119 CX6YD9 89545538 IC50 = 50 nM T12119 CY3H1N 89545616 IC50 = 116 nM T12119 CG7LY8 89545641 IC50 = 171 nM T12119 CK3S4X 89545668 IC50 = 194 nM T12119 CMZ8P5 89545670 IC50 = 130 nM T12119 C74SBC 89555961 IC50 = 76 nM T12119 C01NKB 89555963 IC50 = 71 nM T12119 C29LHS 89556026 IC50 = 7.9 nM T12119 CXHC49 89556028 IC50 = 84 nM T12119 CJRK20 89556063 IC50 = 7 nM T12119 CH6AT7 89556066 IC50 = 32 nM T12119 C9AMI1 89556077 IC50 = 53 nM T12119 CI2T5W 89556108 IC50 = 1889 nM T12119 C51DKP 89556111 IC50 = 23 nM T12119 CK9F0N 89556121 IC50 = 38 nM T12119 C72BSC 89556129 IC50 = 33 nM T12119 CDMI85 89556132 IC50 = 164 nM T12119 CM6SL8 89613863 IC50 = 730 nM T12119 CUB41D 89614421 IC50 = 140 nM T12119 CK8O4U 89614559 IC50 = 810 nM T12119 C90UQK 89614650 IC50 = 150 nM T12119 CQK1S9 89614770 IC50 = 2500 nM T12119 C1HDS6 89683010 IC50 = 100 nM T12119 CV7UN4 89761281 IC50 = 190 nM T12119 C7PT4Z 89761284 IC50 = 250 nM T12119 CAO3I6 89761608 IC50 = 2000 nM T12119 C29BFD 89761642 IC50 = 280 nM T12119 CGI6O0 89761704 IC50 = 520 nM T12119 C8IJ0Y 89761742 IC50 = 140 nM T12119 C4BQC6 89761777 IC50 = 380 nM T12119 COU52N 89761779 IC50 = 120 nM T12119 C2NB6L 89761936 IC50 = 2800 nM T12119 C95IFK 89761981 IC50 = 210 nM T12119 CH6F1I 89963001 IC50 = 2.6 nM T12119 CTKP85 90017371 IC50 = 398.11 nM T12119 C48RCZ 90021555 IC50 = 2.1 nM T12119 C9KH8U 90460903 IC50 = 3880 nM T12119 CXD93Q 90461471 IC50 = 20 nM T12119 CB3YV0 90463221 IC50 = 30 nM T12119 COYC71 90700276 IC50 = 21 nM T12119 CN07GH 90846203 IC50 = 9 nM T12119 CX85KF 91134217 IC50 = 47 nM T12119 C0J3FL 91664339 IC50 = 370 nM T12119 CE76UC 91664340 Ki = 230 nM T12119 C26BZK 91666633 IC50 = 3 nM T12119 C9ETC1 91666645 IC50 = 12 nM T12119 C0S3JN 91799666 IC50 = 10 nM T12119 C7NLE8 91809347 IC50 = 0.4 nM T12119 CTS64R 91809389 IC50 = 30 nM T12119 C6A4OH 91820662 IC50 = 10 nM T12119 C4MB8R 91938052 IC50 = 1 nM T12119 CXN69G 100657083 IC50 = 260 nM T12119 CQO2Y7 100951629 IC50 = 0.1 nM T12119 CHM5W0 117608511 IC50 = 50 nM T12119 C5I2WO 117608537 IC50 = 170 nM T12119 CNFW42 117608566 IC50 = 2 nM T12119 CZX70W 117608604 IC50 = 120 nM T12119 C6O7ZX 117736868 IC50 = 3 nM T12119 CV94EU 117736992 IC50 = 27 nM T12119 CVI38D 117737118 IC50 = 18 nM T12119 CI0D1R 117737120 IC50 = 7 nM T12119 C23NPF 117737172 IC50 = 17 nM T12119 CM1T3I 117737215 IC50 = 11 nM T12119 CN1E5U 117737262 IC50 = 8 nM T12119 CS4IW2 117739617 IC50 = 11 nM T12119 C4NH6M 117740584 IC50 = 37 nM T12119 CFJ97D 117741583 IC50 = 9 nM T12119 CUZ6C2 117741590 IC50 = 270 nM T12119 C0V3KH 117741592 IC50 = 10 nM T12119 CC1A0T 117741702 IC50 = 39 nM T12119 C3C2YG 117741784 IC50 = 120 nM T12119 C4ZO0A 117741876 IC50 = 47 nM T12119 CBL12U 117748926 IC50 = 23 nM T12119 C10BKY 117749324 IC50 = 6 nM T12119 CFV29O 117753901 IC50 = 28 nM T12119 COVX65 117753917 IC50 = 85 nM T12119 CS5X4R 117753922 IC50 = 28 nM T12119 C1OIR7 117753929 IC50 = 61 nM T12119 CQK1U5 117753939 IC50 = 41 nM T12119 CW8RS3 117760464 IC50 = 740 nM T12119 C3P1LN 117789501 IC50 = 41 nM T12119 CK0RV9 117993874 IC50 = 110 nM T12119 CL4O0J 117993881 IC50 = 54 nM T12119 CB8I3S 117993884 IC50 = 62 nM T12119 C92RVJ 117993886 IC50 = 36 nM T12119 CM2H5Q 117993976 IC50 = 28 nM T12119 C9KV7L 117993993 IC50 = 17 nM T12119 CNV24M 117993998 IC50 = 530 nM T12119 C8DSV0 117994021 IC50 = 109 nM T12119 C57PMF 118002063 IC50 = 1190 nM T12119 CT8C0X 118109014 IC50 = 210 nM T12119 COH9J3 118109161 IC50 = 160 nM T12119 CG3M4J 118109168 IC50 = 45 nM T12119 CO6KX7 118109201 IC50 = 27 nM T12119 CAU5T9 118109234 IC50 = 215 nM T12119 CT4ZN7 118109256 IC50 = 112 nM T12119 CG8FJ5 118109302 IC50 = 375 nM T12119 C8OAL5 118109304 IC50 = 30 nM T12119 C3N0KS 118109319 IC50 = 142 nM T12119 CU85FO 118109356 IC50 = 5 nM T12119 CWJ7T6 118109371 IC50 = 12 nM T12119 CS0B7V 118112295 IC50 = 136 nM T12119 CWR6I1 118112300 IC50 = 8 nM T12119 CXY23I 118121135 IC50 = 91 nM T12119 CB4I7H 118121139 IC50 = 44 nM T12119 C7HJ6B 118126600 IC50 = 3500 nM T12119 CF08MJ 118158979 IC50 = 1800 nM T12119 C50RMA 118158981 Ki = 1030 nM T12119 C6ETQ5 118158983 IC50 = 840 nM T12119 C8A6YH 118158984 Ki = 560 nM T12119 CXKV34 118158989 IC50 > 10000 nM T12119 CK4Y1O 118158990 IC50 = 2570 nM T12119 CE7K1A 118158995 Ki = 920 nM T12119 C92NSO 118158996 Ki = 650 nM T12119 C2G6VY 118158998 Ki = 3030 nM T12119 C31XNM 118193882 IC50 = 2360 nM T12119 CHSB45 118193883 IC50 = 90 nM T12119 CWAI23 118193935 IC50 = 150 nM T12119 C50DIN 118193948 IC50 = 60 nM T12119 CU20DG 118193996 IC50 = 400 nM T12119 CCN3J9 118255610 IC50 > 20000 nM T12119 C9WR4Y 118255620 IC50 = 340 nM T12119 CS9IW6 118255624 Ki = 630 nM T12119 CW6M2K 118255632 IC50 = 400 nM T12119 CM7D9K 118255633 IC50 = 360 nM T12119 CA74UH 118255641 IC50 = 670 nM T12119 C27ZAP 118255642 Ki = 440 nM T12119 C2Z0EY 118255648 IC50 = 910 nM T12119 CTF16A 118255649 Ki = 450 nM T12119 CD3E1A 118255663 IC50 = 1920 nM T12119 C7RZL3 118255664 Ki = 300 nM T12119 C7P0GN 118255669 Ki = 550 nM T12119 CU0Q2O 118255675 IC50 = 580 nM T12119 CTV4D2 118267016 Ki = 400 nM T12119 CF23UM 118267018 Ki = 300 nM T12119 C0U9RS 118418144 IC50 = 9 nM T12119 C4Y7CV 118418152 IC50 = 13 nM T12119 C8RUX7 118418168 IC50 = 9 nM T12119 C7JRN5 118418195 IC50 = 2 nM T12119 C0L3QA 118418208 IC50 = 4 nM T12119 CQX2I8 118418217 IC50 = 2 nM T12119 CJS7U3 118418225 IC50 = 8 nM T12119 C1G2LI 118418233 IC50 = 4 nM T12119 CU3I7E 118418380 IC50 = 9 nM T12119 C4GVZ5 118418435 IC50 = 4 nM T12119 CQ3WK8 118540765 IC50 = 1.5 nM T12119 C7AYV5 118540795 IC50 = 0.01 nM T12119 CG5O4Q 118540838 IC50 < 4 nM T12119 CKA2F8 118554582 IC50 < 10 nM T12119 CE1JG2 118653870 IC50 = 13 nM T12119 CG51WM 118657693 IC50 = 1180 nM T12119 CR8TX9 118708662 IC50 = 0.3 nM T12119 CN0K2R 118708663 IC50 = 423 nM T12119 C6M2XV 118708664 IC50 = 0.2 nM T12119 CBA2R3 118708665 IC50 = 1.7 nM T12119 CJ6O2Z 118708666 IC50 = 1 nM T12119 C9YPR6 118708667 IC50 = 552 nM T12119 C7J4GA 118708668 IC50 = 1 nM T12119 CHV68E 118708669 IC50 = 4 nM T12119 CF93GI 118708670 IC50 = 3 nM T12119 CWE7O3 118708671 IC50 = 5 nM T12119 CTW3E0 118708672 IC50 = 67 nM T12119 C9BM3K 118708673 IC50 = 8 nM T12119 C1R5WS 118708674 IC50 = 10 nM T12119 CDJR23 118708675 IC50 = 18 nM T12119 C85DXB 118708676 IC50 = 528 nM T12119 CR7HG8 118708677 IC50 = 0.23 nM T12119 C17PGH 118708678 IC50 = 0.042 nM T12119 CSEC16 118708679 IC50 = 0.6 nM T12119 CDGF38 118708680 IC50 = 0.8 nM T12119 CU9W5V 118708681 IC50 = 293 nM T12119 CG34QX 118708682 IC50 > 3000 nM T12119 CMDN36 118710321 IC50 = 201 nM T12119 CPL32R 118710322 IC50 = 9279 nM T12119 CA79ZM 118710323 IC50 = 8732 nM T12119 CLS68B 118710324 IC50 = 56 nM T12119 CL2PK9 118710325 IC50 = 439 nM T12119 CDO95Z 118710326 IC50 = 9 nM T12119 CG7X9J 118710327 IC50 = 37 nM T12119 C83LIE 118710328 IC50 = 87 nM T12119 CH29DT 118711022 IC50 = 280 nM T12119 C3BQM2 118714771 IC50 = 19 nM T12119 CPVC71 118714772 IC50 = 22 nM T12119 CEB6T7 118714773 IC50 = 63 nM T12119 C65NKL 118714774 IC50 = 80 nM T12119 C39NSR 118714775 IC50 = 315 nM T12119 CJ8E7U 118714776 IC50 = 103 nM T12119 C84KNW 118714777 IC50 = 5723 nM T12119 CHS5K3 118714778 IC50 = 656 nM T12119 C58YHZ 118714779 IC50 = 439 nM T12119 CF2YQ4 118714780 IC50 = 15200 nM T12119 C40SOZ 118714781 IC50 = 106 nM T12119 C67FSV 118714782 IC50 = 73 nM T12119 CREM47 118714783 IC50 = 124 nM T12119 CX4I5Q 118714784 IC50 = 73 nM T12119 C5YWC2 118716175 Ki = 27 nM T12119 CH96JD 118716176 IC50 = 620 nM T12119 C69PLO 118734433 IC50 = 370 nM T12119 C2NAE8 118734434 IC50 = 100 nM T12119 CD4B5E 118734435 IC50 = 430 nM T12119 C91PCO 118734436 IC50 = 270 nM T12119 CM2Y6W 118734437 IC50 = 13.2 nM T12119 CFL60J 118734438 IC50 = 430 nM T12119 CQ0R3E 118734439 IC50 = 940 nM T12119 CY8A1T 118734440 IC50 = 500 nM T12119 CFRZ45 118734441 IC50 = 210 nM T12119 C3ZJ0K 118734442 IC50 = 170 nM T12119 CI30YK 118734443 IC50 = 120 nM T12119 CUAQ60 118734444 IC50 = 190 nM T12119 CFNR84 118734445 IC50 = 230 nM T12119 CK12TX 118734446 IC50 = 130 nM T12119 C09BDT 118734447 IC50 = 90 nM T12119 C6F9BI 118734448 IC50 = 690 nM T12119 C8ZLX9 118734449 IC50 = 190 nM T12119 C01BNE 118734450 IC50 = 380 nM T12119 CI0FE2 118734451 IC50 = 470 nM T12119 C1CED0 118734452 IC50 = 330 nM T12119 C8NBL5 118734453 IC50 = 260 nM T12119 C0CY2K 118734454 IC50 = 970 nM T12119 CTR7O8 118734455 IC50 = 470 nM T12119 CZQD84 118734456 IC50 > 5000 nM T12119 CGBF25 118734457 IC50 > 5000 nM T12119 C6I8HF 118734458 IC50 = 800 nM T12119 C5G7DQ 118734459 IC50 = 170 nM T12119 CVW15D 118734460 IC50 = 1200 nM T12119 CSE60C 118734461 IC50 = 410 nM T12119 CO4U1R 118734462 IC50 = 9 nM T12119 CA95IF 118734463 IC50 = 79 nM T12119 C14ILF 118734464 IC50 = 39 nM T12119 C3TOV9 118734465 IC50 = 19 nM T12119 C2RO8T 118734466 IC50 = 2 nM T12119 CSP25D 118734467 IC50 = 9 nM T12119 CJD80C 118734468 IC50 = 5 nM T12119 C06TAI 118734469 IC50 = 25 nM T12119 CBY5M0 118734470 IC50 = 24 nM T12119 CHO8I3 118734471 IC50 = 4 nM T12119 C38BCH 118734472 IC50 = 5 nM T12119 CV7UH5 118734473 IC50 = 6 nM T12119 C6SEA7 118734474 IC50 = 236 nM T12119 CO7DP2 118734475 IC50 = 86 nM T12119 CX2R0E 118734476 IC50 = 8 nM T12119 C16AEK 118734477 IC50 = 24 nM T12119 CO1UF9 118734478 IC50 = 4 nM T12119 C16AUM 118734479 IC50 = 19 nM T12119 CI2P1V 118734480 IC50 = 63 nM T12119 C1Z8AN 118734481 IC50 = 23 nM T12119 CYD8N6 118734482 IC50 = 7 nM T12119 CW05LY 118734483 IC50 = 10 nM T12119 CN01US 118734484 IC50 = 28 nM T12119 C3E7GP 118734485 IC50 = 13 nM T12119 CCA41Z 118734486 IC50 = 59 nM T12119 CM2QS5 118734487 IC50 = 3 nM T12119 C3T1QC 118734488 IC50 = 4 nM T12119 CM6Y8X 118734489 IC50 = 5 nM T12119 C93LMC 118734490 IC50 = 34 nM T12119 C8LHA3 118734491 IC50 = 4 nM T12119 C26ADB 118734547 IC50 = 8 nM T12119 C82UBF 118734548 IC50 = 29 nM T12119 CO4KD2 118734549 IC50 = 54 nM T12119 CX6L4C 118734550 IC50 = 4 nM T12119 C5JNX2 118734551 IC50 = 11 nM T12119 C0UJ8Q 118734552 IC50 = 8 nM T12119 CJDP52 118734553 IC50 = 1.6 nM T12119 C0RFQ5 118937646 IC50 = 1500 nM T12119 CTR37C 118937656 IC50 = 270 nM T12119 CTC20B 118937664 IC50 = 840 nM T12119 CR9Y6M 118937702 IC50 = 330 nM T12119 C1Y7MU 118937716 IC50 = 1100 nM T12119 C9JL4Y 118937760 IC50 = 370 nM T12119 C8JEV3 118937784 IC50 = 9000 nM T12119 CXI1F9 118937849 IC50 = 920 nM T12119 CWL1S3 118937903 IC50 = 810 nM T12119 CXZ43S 118937913 IC50 = 730 nM T12119 CMQB61 118937925 IC50 = 570 nM T12119 CHQ7J9 118937930 IC50 = 900 nM T12119 C9H0BR 121333853 IC50 = 220 nM T12119 CGH4B7 121333855 IC50 = 68 nM T12119 CZ3X9J 121333858 IC50 = 60 nM T12119 C4XRZ6 121333863 IC50 = 170 nM T12119 CT4FA9 121333871 IC50 = 37 nM T12119 CIQ8C0 121333899 IC50 = 40 nM T12119 C83STC 121333902 IC50 = 140 nM T12119 CMA2O3 121333930 IC50 = 120 nM T12119 C9Q2ND 121333973 IC50 = 17 nM T12119 C7W0AX 122190006 IC50 = 21 nM T12119 CHPL50 122194669 IC50 = 1000 nM T12119 CWSA14 122194670 IC50 = 500 nM T12119 C05AUF 122194671 IC50 = 480 nM T12119 CY2B6W 122194672 IC50 = 1100 nM T12119 CP38IW 122194673 IC50 = 1200 nM T12119 CWGY65 122194675 IC50 = 700 nM T12119 C1MH8Y 122194676 IC50 = 1000 nM T12119 CP4L5A 122194677 IC50 = 1700 nM T12119 CW3D9H 122196008 IC50 = 3900 nM T12119 C5G9FH 122196009 IC50 = 780 nM T12119 C2RBF4 122196010 IC50 = 3700 nM T12119 C0R8OS 122196011 IC50 = 1300 nM T12119 C61QNK 122196012 IC50 = 24000 nM T12119 CZ2HR6 122196013 IC50 = 1100 nM T12119 C6W5IA 122196014 IC50 = 1800 nM T12119 CKEH54 122196015 IC50 = 9400 nM T12119 C38XFL 122196016 IC50 = 1500 nM T12119 CLQ8O5 122196017 IC50 = 1100 nM T12119 C82UNL 122196018 IC50 = 1200 nM T12119 C0KG7Z 122196019 IC50 = 900 nM T12119 CS0W4O 122196020 IC50 = 380 nM T12119 CK8FH3 122196021 IC50 = 3400 nM T12119 C9N1CF 122196022 IC50 = 5300 nM T12119 CR4JT9 122196023 IC50 = 1400 nM T12119 C80OZQ 122196024 IC50 = 1800 nM T12119 CT9N7O 122196025 IC50 = 2800 nM T12119 C3B0RY 122422350 IC50 = 88 nM T12119 C81EPB 122422402 IC50 = 100 nM T12119 CC2TE4 122422536 IC50 = 77 nM T12119 C2ON8G 122458653 IC50 = 39 nM T12119 CEGS87 122513481 IC50 = 1350 nM T12119 C9K5RV 122513516 IC50 = 340 nM T12119 CC1J0T 122591381 IC50 = 240 nM T12119 CA3S8B 124221798 IC50 = 10 nM T12119 C3I0PD 124221800 IC50 = 22 nM T12119 CVKO13 124221803 IC50 = 7.3 nM T12119 CVI8X5 124221907 IC50 = 69 nM T12119 C84FIJ 124221975 IC50 = 5 nM T12119 C01UFA 124221976 IC50 = 7 nM T12119 CEC9K6 127030665 IC50 = 5 nM T12119 C5EGJ8 127034190 IC50 = 4 nM T12119 CL8H5W 127034191 IC50 = 14 nM T12119 C7JT8V 127045799 IC50 = 2.3 nM T12119 CH2Z3S 127045806 IC50 = 120 nM T12119 CSJD60 127045808 IC50 = 280 nM T12119 COWD91 127045811 IC50 = 33 nM T12119 C90JPN 127045813 IC50 > 5000 nM T12119 C21JCE 127045825 IC50 = 590 nM T12119 CNF0G1 127045829 IC50 = 1400 nM T12119 CC9TY3 127045830 IC50 = 150 nM T12119 CDC0M9 127046018 IC50 = 50 nM T12119 C74SHI 127046022 IC50 = 380 nM T12119 CH0CD1 127046023 IC50 = 1500 nM T12119 CPX1F0 127046025 IC50 > 4900 nM T12119 CAVD37 127046026 IC50 = 540 nM T12119 C8UW6X 127046032 IC50 = 250 nM T12119 CMPZ51 127046033 IC50 = 50 nM T12119 CY5J0R 127046039 IC50 = 230 nM T12119 CBQ47D 127046045 IC50 = 630 nM T12119 C6NVQ1 127046047 IC50 = 590 nM T12119 C4MU2J 127046230 IC50 = 70 nM T12119 CGYE23 127046231 IC50 = 860 nM T12119 C69GBJ 127046239 IC50 = 200 nM T12119 CM1IH3 127046241 IC50 = 130 nM T12119 C4L1VA 127046242 IC50 = 320 nM T12119 CWN2J7 127046243 IC50 = 6 nM T12119 CI1VA2 127046252 IC50 = 1.6 nM T12119 CE67AD 127046253 IC50 = 4 nM T12119 C53RIX 127046257 IC50 = 970 nM T12119 COK9Z3 127046259 IC50 = 70 nM T12119 CL5VY9 127046359 IC50 = 5 nM T12119 C3M6YT 127046415 IC50 = 190 nM T12119 C90HYR 127046420 IC50 = 80 nM T12119 C8BES0 127046422 IC50 = 5 nM T12119 C2EI4Q 127046423 IC50 = 16 nM T12119 CM2HB0 127046424 IC50 = 30 nM T12119 CM5D6J 127046425 IC50 = 50 nM T12119 C9LH4U 127046428 IC50 = 2350 nM T12119 C20KGH 127046429 IC50 = 100 nM T12119 CH27MP 127046433 IC50 > 5000 nM T12119 CWH7Y0 127046434 IC50 > 5000 nM T12119 C1CV8E 127046436 IC50 = 110 nM T12119 C87YLU 127046583 IC50 > 5000 nM T12119 C74ELB 127046587 IC50 = 80 nM T12119 CI9XY7 127046589 IC50 = 280 nM T12119 CQ3EV4 127046592 IC50 = 220 nM T12119 C8PO4C 127046597 IC50 = 4 nM T12119 C31XHN 127046598 IC50 = 40 nM T12119 CFSH84 127046606 IC50 = 120 nM T12119 CP8T2D 127046764 IC50 = 50 nM T12119 C0A7SK 127046767 IC50 = 260 nM T12119 CC2Y1J 127046770 IC50 = 3500 nM T12119 C1XON9 127046774 IC50 = 1400 nM T12119 C80RLU 127046781 IC50 > 5000 nM T12119 C34GAN 127046799 IC50 = 1100 nM T12119 CS0M4H 127046800 IC50 = 320 nM T12119 CV09PX 127046801 IC50 = 2600 nM T12119 CCXR80 127046802 IC50 = 2000 nM T12119 CJRV57 127046803 IC50 = 3800 nM T12119 COG64J 127046804 IC50 = 580 nM T12119 CSKX63 127046908 IC50 = 18 nM T12119 CVUW94 127046909 IC50 = 42 nM T12119 C02HPV 127046912 IC50 = 50 nM T12119 C8CK6P 127046914 IC50 = 1750 nM T12119 C3CSI0 127046916 IC50 = 3 nM T12119 C4X2OU 127046919 IC50 = 260 nM T12119 CL9W8T 127046920 IC50 = 60 nM T12119 CLH51Y 127046923 IC50 > 5000 nM T12119 CXMC23 127046930 IC50 > 5000 nM T12119 CB9EF5 127046932 IC50 = 110 nM T12119 CZ7G6T 127047057 IC50 = 220 nM T12119 CND20E 127047062 IC50 = 4 nM T12119 CNSZ83 127047063 IC50 = 270 nM T12119 C1R4VN 127047068 IC50 > 5000 nM T12119 C5VU7H 127047069 IC50 = 220 nM T12119 CFG94A 127047073 IC50 = 3600 nM T12119 CF5D0S 127047074 IC50 > 4900 nM T12119 C0XS7B 127047075 IC50 = 2350 nM T12119 CI60KD 127047206 IC50 = 12 nM T12119 CA7YG4 127047208 IC50 > 5000 nM T12119 CXT5Y0 127047216 IC50 = 100 nM T12119 CY8RH9 127047220 IC50 > 5000 nM T12119 CV4OB1 127047223 IC50 = 200 nM T12119 C1RD6X 127047251 IC50 = 190 nM T12119 CZLT12 127047252 IC50 = 580 nM T12119 CFPJ73 127047320 IC50 > 5000 nM T12119 C3JK6P 127047322 IC50 = 170 nM T12119 C1T5PC 127047323 IC50 = 2.1 nM T12119 C28REX 127047327 IC50 = 110 nM T12119 CVSF19 127047330 IC50 = 130 nM T12119 C0IO2K 127047331 IC50 = 200 nM T12119 C9SIK3 127047333 IC50 = 170 nM T12119 CKD78E 127047346 IC50 = 50 nM T12119 C5DO7I 127047347 IC50 = 110 nM T12119 CM5TX2 127047468 IC50 > 5000 nM T12119 C54TRJ 127047469 IC50 = 100 nM T12119 C3K5YI 127047471 IC50 = 220 nM T12119 C2M5JH 127047472 IC50 = 170 nM T12119 C3SLJ4 127047473 IC50 = 100 nM T12119 CCA51M 127047474 IC50 = 2 nM T12119 C6EM0G 127047476 IC50 = 720 nM T12119 C5RKB7 127047479 IC50 = 120 nM T12119 C96VDX 127047480 IC50 = 90 nM T12119 CJ7IQ4 127047485 IC50 = 40 nM T12119 CZKB91 127047487 IC50 = 280 nM T12119 C7OTX3 127047488 IC50 = 80 nM T12119 CVR95B 127047489 IC50 = 140 nM T12119 CW8P5Y 127047613 IC50 = 210 nM T12119 C0WXP3 127047615 IC50 = 12 nM T12119 C1RK5C 127047619 IC50 > 4900 nM T12119 C9QZH7 127047622 IC50 = 6 nM T12119 CJ31BC 127047628 IC50 = 560 nM T12119 C9MXK5 127047633 IC50 = 70 nM T12119 CB16MW 127047643 IC50 = 1400 nM T12119 C7HQV4 127047644 IC50 = 110 nM T12119 C09QIY 127047645 IC50 = 1900 nM T12119 C5S1AI 127047646 IC50 = 960 nM T12119 C1ULZ3 127047735 IC50 = 180 nM T12119 C4T5WS 127047736 IC50 = 950 nM T12119 CQ45AO 127047757 IC50 = 140 nM T12119 CG5X0Y 127047758 IC50 = 8 nM T12119 CTRE63 127047854 IC50 = 1500 nM T12119 CDGS14 127047866 IC50 = 4450 nM T12119 C16NUB 127047867 IC50 = 80 nM T12119 CG52RP 127047873 IC50 = 130 nM T12119 C8PWL6 127047983 IC50 = 1030 nM T12119 CGW63M 127047988 IC50 = 60 nM T12119 CR6AB0 127047989 IC50 > 5000 nM T12119 CK9ZO8 127047990 IC50 = 140 nM T12119 CQ2SO8 127047999 IC50 = 1.9 nM T12119 C2D9LN 127048108 IC50 = 2.5 nM T12119 C25GJD 127048113 IC50 = 30 nM T12119 C4VID9 127048115 IC50 = 470 nM T12119 CCI81A 127048120 IC50 = 270 nM T12119 CE1Z4W 127048121 IC50 = 90 nM T12119 CI0P1M 127048127 IC50 = 80 nM T12119 C4CUP9 127048128 IC50 = 70 nM T12119 C7HGD0 127048130 IC50 = 6 nM T12119 C4LK6A 127048137 IC50 = 1700 nM T12119 CNA30T 127048138 IC50 = 1.9 nM T12119 C1WAE8 127050785 IC50 = 241 nM T12119 C0M4AK 127050786 IC50 = 5200 nM T12119 CA35IE 130454905 IC50 = 15 nM T12119 C5KWH0 132020346 IC50 = 790 nM T12119 C4A2JF 132020399 IC50 = 82 nM T12119 C9C5PT 132020406 IC50 = 164 nM T12119 COH0K2 132020407 IC50 > 3000 nM T12119 CX6WL3 132020408 IC50 = 740 nM T12119 CABH81 132020419 IC50 = 91 nM T12119 C79BLN 132020421 IC50 = 1300 nM T12119 CDN3E8 132020424 IC50 = 4200 nM T12119 CZ5H2B 132020452 IC50 = 8 nM T12119 CNK15D 132020464 IC50 = 530 nM T12119 CMD5X6 132020466 IC50 = 460 nM T12119 C4FPR1 132020468 IC50 = 262 nM T12119 CTRG94 132020475 IC50 = 69 nM T12119 C76RHU 132020480 IC50 = 600 nM T12119 C6ME9R 132020486 IC50 = 3330 nM T12119 C69ELN 132020488 IC50 = 700 nM T12119 CIM31O 132020491 IC50 = 154 nM T12119 CB74IC 132020507 IC50 = 290 nM T12119 C4JP3T 132020512 IC50 = 380 nM T12119 CDL95F 132020518 IC50 = 88 nM T12119 CUZ03K 132020526 IC50 = 38 nM T12119 CD4HS0 132020533 IC50 = 420 nM T12119 C5LYQ6 132020541 IC50 = 13 nM T12119 C5G1PQ 132020544 IC50 = 8 nM T12119 CAZI64 132020570 IC50 = 19 nM T12119 CTC7E3 132020571 IC50 = 66 nM T12119 CP8A1Q 132020575 IC50 = 89 nM T12119 C7ZIP5 132020580 IC50 = 810 nM T12119 CLV79P 132020582 IC50 = 3.3 nM T12119 CF2QM1 132020584 IC50 = 1.1 nM T12119 CR92US 132020585 IC50 = 1300 nM T12119 CJVH59 132020588 IC50 = 123 nM T12119 CM42HK 132020589 IC50 = 220 nM T12119 C21QHW 132051336 IC50 = 80 nM T12119 C9RBP0 132051461 IC50 = 740 nM T12119 CVFK13 132051462 IC50 = 23 nM T12119 CNCO16 132051469 IC50 = 190 nM T12119 CEHO59 132051625 IC50 = 1420 nM T12119 CNZA27 132051626 IC50 = 170 nM T12119 CHL97M 132051650 IC50 = 8100 nM T12119 C83UBM 132051677 IC50 = 16 nM T12119 CF2M4S 134132899 IC50 = 1400 nM T12119 C1M8ZR 134133921 IC50 = 1500 nM T12119 CX3R6G 134134034 IC50 = 7 nM T12119 CPV1K0 134134546 IC50 = 3.2 nM T12119 CIZ4N6 134138462 IC50 = 23.7 nM T12119 CM2FJ0 134140349 IC50 = 2.8 nM T12119 C62IUH 134140917 IC50 = 6.7 nM T12119 CI2DB0 134141246 IC50 > 30000 nM T12119 C5LU2O 134142620 IC50 = 12.3 nM T12119 CBN9M8 134145535 IC50 = 2.3 nM T12119 CN7RI4 134146511 IC50 = 37 nM T12119 CYW3K5 134146818 IC50 = 1.3 nM T12119 C9BX7F 134147105 IC50 = 4.3 nM T12119 CC51AX 134148459 IC50 = 4 nM T12119 CIJ1R2 134150038 IC50 = 28.1 nM T12119 CV5Q7F 134150730 IC50 = 1.3 nM T12119 CA58DN 134152190 IC50 = 4.7 nM T12119 C8I6FX 134153393 IC50 = 15.2 nM T12119 C1S8IQ 134153460 IC50 = 5.5 nM T12119 CS5ZV8 134155845 IC50 > 30000 nM T12119 CK6O0G 134156125 IC50 = 19.6 nM T12119 CJQ94D 134201162 IC50 = 33 nM T12119 CIW86J 134429539 IC50 = 38 nM T12119 CFYC29 134477061 IC50 = 29 nM T12119 C20QBE 134477062 IC50 = 4 nM T12119 CT58HM 134477070 IC50 = 15 nM T12119 C32HVP 134477090 IC50 = 15 nM T12119 CAED75 134477093 IC50 = 339 nM T12119 CO15IT 134477094 IC50 = 70 nM T12119 CH27DQ 134477104 IC50 = 78 nM T12119 C0Q1MD 134477108 IC50 = 78 nM T12119 CX64SG 134477133 IC50 = 105 nM T12119 CT7J4U 134477136 IC50 = 14 nM T12119 C03SFG 134477143 IC50 = 17 nM T12119 C70XMC 134477147 IC50 = 42 nM T12119 CL06KE 134477148 IC50 = 8.4 nM T12119 C7JM1E 134477177 IC50 = 11 nM T12119 C4LS2A 134477178 IC50 = 16 nM T12119 C9WN3E 134477214 IC50 = 8 nM T12119 C9IB8P 134477217 IC50 = 69 nM T12119 CN37XZ 134477224 IC50 = 64 nM T12119 CR39TS 134477260 IC50 = 9 nM T12119 CWNK85 134477261 IC50 = 12 nM T12119 C1R9DV 134477283 IC50 = 10 nM T12119 CJ3X7K 135283936 IC50 = 15.3 nM T12119 C3QBM8 135284018 Ki > 700 nM T12119 CN1E2Q 135284025 Ki = 0.85 nM T12119 CL62WI 135284073 Ki > 700 nM T12119 CWU9I0 135284152 Ki = 509 nM T12119 CBE1T5 135284349 IC50 = 0.57 nM T12119 C12XAW 135356858 IC50 = 87 nM T12119 C27POJ 135356894 IC50 = 50 nM T12119 C13VUE 135356902 IC50 = 7.6 nM T12119 CMH4G1 135412290 IC50 = 940 nM T12119 CVY28Z 135412524 IC50 = 20000 nM T12119 CB1VD9 135426471 IC50 = 680 nM T12119 C1MVP9 135427582 IC50 > 30000 nM T12119 CQ68EK 135439429 IC50 = 5400 nM T12119 C7DR4L 135442530 IC50 = 4700 nM T12119 CY1N4E 135480550 IC50 = 1300 nM T12119 CRBQ97 135481198 IC50 > 30000 nM T12119 C2Q7WG 135496350 IC50 > 30000 nM T12119 CO7XF5 135537663 IC50 = 950 nM T12119 CMO04Z 135926523 IC50 = 340 nM T12119 C2JW5S 135981385 IC50 > 30000 nM T12119 CN13KF 136042279 IC50 = 3200 nM T12119 C6MZD2 136042280 IC50 = 2200 nM T12119 CZVG23 136042281 IC50 > 30000 nM T12119 CLHZ61 136042282 IC50 = 1200 nM T12119 CZ68AW 136042283 IC50 = 2500 nM T12119 C6IJV1 136042284 IC50 = 7800 nM T12119 CM2C9X 136042285 IC50 > 30000 nM T12119 CB50TE 136042286 IC50 = 4300 nM T12119 CJ64ZH 136042287 IC50 > 30000 nM T12119 CKF7M8 136042288 IC50 > 30000 nM T12119 CN3HU2 136180780 IC50 = 130 nM T12119 CVFN62 136180781 IC50 = 260 nM T12119 C1RSX2 136180782 IC50 = 300 nM T12119 C0MIN5 137631475 IC50 = 1030 nM T12119 C8JA9G 137631733 IC50 = 264 nM T12119 C2XI8Y 137632393 IC50 = 8 nM T12119 CNGF31 137632548 IC50 = 70 nM T12119 C3X8OM 137633120 IC50 = 170 nM T12119 C4RNK9 137633146 IC50 = 640 nM T12119 C2Z4RA 137633695 IC50 = 160 nM T12119 CJ8R5B 137634460 IC50 = 90 nM T12119 CLG25H 137634494 IC50 = 815 nM T12119 C1VI7A 137634947 IC50 = 340 nM T12119 C4LXK8 137636188 IC50 = 23 nM T12119 C08DOT 137636231 IC50 = 48 nM T12119 CU8Z4V 137636977 IC50 = 70 nM T12119 CKI1P5 137637043 IC50 = 50 nM T12119 CUP6F0 137637379 IC50 = 50 nM T12119 CK60TZ 137637389 IC50 = 90 nM T12119 CO3QJ8 137637393 IC50 = 43 nM T12119 C90PYH 137637423 IC50 = 3100 nM T12119 CE46QO 137637515 IC50 = 40 nM T12119 CJH2V9 137637559 IC50 = 8700 nM T12119 C5YV3A 137637566 IC50 = 57 nM T12119 CEN8M3 137638107 IC50 = 1800 nM T12119 CW95QX 137638418 IC50 = 150 nM T12119 CEP37F 137638536 IC50 = 970 nM T12119 C0ZS9N 137638993 IC50 = 78 nM T12119 C0FCQ3 137639043 IC50 > 25000 nM T12119 CJ91IS 137639164 IC50 = 80 nM T12119 CZ2A5K 137639461 IC50 = 207 nM T12119 CMR69P 137639538 IC50 = 60 nM T12119 CIZ75D 137639905 IC50 = 420 nM T12119 CK1C5F 137640087 IC50 = 47 nM T12119 CA2Z1P 137640897 IC50 = 900 nM T12119 CP2IO8 137640927 IC50 = 440 nM T12119 CIF8C5 137641071 IC50 = 1700 nM T12119 C3DB7L 137641284 IC50 = 130 nM T12119 C23OFG 137641349 IC50 = 80 nM T12119 CT68NG 137641840 IC50 = 90 nM T12119 CMG4L2 137642297 IC50 = 20 nM T12119 CPW7T0 137643121 IC50 = 11 nM T12119 CMN61F 137644207 IC50 = 590 nM T12119 CSK75M 137644331 IC50 = 250 nM T12119 CM8HD7 137644363 IC50 > 10000 nM T12119 CQB6Z2 137644815 IC50 = 3900 nM T12119 CND2Z9 137645152 IC50 = 1700 nM T12119 CL3F2Y 137645273 IC50 = 780 nM T12119 C9HCP2 137645311 IC50 = 80 nM T12119 CE6GN1 137645760 IC50 = 1450 nM T12119 CJYG62 137645851 IC50 = 70 nM T12119 C9Q0MH 137645867 IC50 = 12 nM T12119 C89NAZ 137646053 IC50 = 40 nM T12119 CFKR53 137646837 IC50 = 49 nM T12119 C4XVD2 137647076 IC50 = 16 nM T12119 C9L8CZ 137647771 IC50 = 61 nM T12119 CD2WA1 137647899 IC50 = 150 nM T12119 CIYO97 137647989 IC50 = 90 nM T12119 C3VO8H 137648536 IC50 = 510 nM T12119 CQ8E6R 137649015 IC50 = 4300 nM T12119 CQ93EC 137649075 IC50 = 18 nM T12119 CYB94V 137649148 IC50 = 900 nM T12119 CV03MT 137649269 IC50 = 20 nM T12119 CJ59RF 137649283 IC50 = 66 nM T12119 C04JSE 137649716 IC50 = 24 nM T12119 C8N9CH 137650363 IC50 = 13 nM T12119 C6PL9C 137651460 IC50 = 16 nM T12119 CUY5V2 137651963 IC50 = 3920 nM T12119 CE1OC6 137651969 IC50 = 7 nM T12119 C1KL5S 137652510 IC50 > 25000 nM T12119 CH5L7O 137652616 IC50 > 10000 nM T12119 CPU9R2 137653152 IC50 = 580 nM T12119 CK14LN 137653163 IC50 = 186 nM T12119 CM1CP2 137653473 IC50 = 490 nM T12119 C3QAT7 137654032 IC50 = 4800 nM T12119 CMJ0X9 137654527 IC50 = 129 nM T12119 CZK41F 137654701 IC50 = 700 nM T12119 C3O2MS 137654877 IC50 = 580 nM T12119 C5FAI1 137654893 IC50 = 250 nM T12119 C5FRH3 137655495 IC50 = 70 nM T12119 C9PJC3 137655604 IC50 = 240 nM T12119 C08ZUM 137657123 IC50 = 3920 nM T12119 C2ME3D 137657693 IC50 = 220 nM T12119 CA72YP 137658615 IC50 = 11 nM T12119 CDO4F5 137658625 IC50 = 54 nM T12119 C5S8BG 137658700 IC50 = 90 nM T12119 CJ8L1W 137659170 IC50 = 31 nM T12119 CZ2G4H 137659479 IC50 = 324 nM T12119 C0Q7VH 137659493 IC50 = 40 nM T12119 C8UK1W 137659739 IC50 = 38 nM T12119 CX32CH 137660496 IC50 = 1670 nM T12119 CU96IH 137660539 IC50 = 80 nM T12119 C2KX3V 137661020 IC50 = 17700 nM T12119 COR59Z 137661415 IC50 = 80 nM T12119 CAJ7S9 137661575 IC50 = 39 nM T12119 CEN5X3 137661781 IC50 = 1540 nM T12119 CJ28FI 138393286 Ki = 0.79 nM T12119 CJ68PM 138558077 IC50 = 2900 nM T12119 CVIC01 138558093 IC50 > 3000 nM T12119 CF78ZM 138571094 IC50 = 1700 nM T12119 CR23HX 145948497 IC50 = 33 nM T12119 CNSU46 145948687 IC50 = 370 nM T12119 CRH94T 145948711 IC50 = 430 nM T12119 CDZK19 145948712 IC50 = 450 nM T12119 C8KW9F 145948730 IC50 = 10 nM T12119 CQPL31 145948977 IC50 = 670 nM T12119 CVJ24I 145949342 IC50 = 22 nM T12119 C38OXE 145949375 IC50 = 71 nM T12119 CVT3Q9 145949606 IC50 = 12.6 nM T12119 CLD04E 145949796 IC50 = 5.7 nM T12119 C5K7VF 145950190 IC50 = 0.5 nM T12119 C7V3HY 145950505 IC50 = 19 nM T12119 C23MIU 145951388 IC50 = 182 nM T12119 C3IPL7 145951679 IC50 = 1.6 nM T12119 C23NCA 145951748 IC50 = 3.1 nM T12119 C7JO8W 145951923 IC50 = 471 nM T12119 C7V2HA 145952303 IC50 = 0.3 nM T12119 C5A2SE 145952369 IC50 = 24 nM T12119 CCR2Y5 145952753 IC50 = 1.7 nM T12119 CR95FI 145953073 IC50 = 22 nM T12119 C8W0LQ 145953367 IC50 = 1.1 nM T12119 CHV56N 145953458 IC50 = 0.6 nM T12119 CRT63U 145953831 IC50 = 1.3 nM T12119 CVBI85 145954213 IC50 = 3 nM T12119 CE3B1L 145954936 IC50 = 8.3 nM T12119 CF6L8Q 145955101 IC50 = 0.26 nM T12119 CQL27G 145955229 IC50 = 1 nM T12119 CSX5K2 145955231 IC50 = 0.6 nM T12119 CA10ZE 145956186 IC50 = 32 nM T12119 CTW9Q4 145956356 IC50 = 0.3 nM T12119 C8NH1M 145957393 IC50 = 8.9 nM T12119 CA5LD6 145957425 IC50 = 540 nM T12119 C80WHY 145957835 IC50 > 1000 nM T12119 CA03MX 145957880 IC50 = 1 nM T12119 CL59SC 145958162 IC50 = 1.3 nM T12119 CVX4N1 145958248 IC50 = 0.2 nM T12119 CCTB54 145958837 IC50 = 0.8 nM T12119 C7Y0MC 145959040 IC50 = 15 nM T12119 C38DYW 145959291 IC50 = 0.5 nM T12119 CDW83O 145959527 IC50 = 2.5 nM T12119 CHX92D 145960265 IC50 = 0.2 nM T12119 CHLT37 145960279 IC50 = 825 nM T12119 CDA42P 145960383 IC50 = 9500 nM T12119 C3PA1D 145960602 IC50 = 190 nM T12119 CM0BG7 145961271 IC50 = 4300 nM T12119 CBHA12 145961383 IC50 = 580 nM T12119 CSAR89 145961545 IC50 = 520 nM T12119 C90GVK 145961619 IC50 = 70 nM T12119 CID6G8 145961739 IC50 = 8900 nM T12119 CRQ9Z2 145962160 IC50 = 149 nM T12119 C5QRS1 145962458 IC50 = 2900 nM T12119 C5HE2I 145962668 IC50 = 100 nM T12119 CWL65X 145962677 IC50 = 940 nM T12119 C52VFR 145962752 IC50 = 170 nM T12119 CS86IX 145963060 IC50 = 800 nM T12119 CP9TU4 145963182 IC50 = 78 nM T12119 C3UZX8 145963617 IC50 = 310 nM T12119 CQT0L8 145963819 IC50 = 310 nM T12119 CQ7Y1N 145963931 IC50 = 1100 nM T12119 C62MVS 145964029 IC50 = 33 nM T12119 C91CMS 145964520 IC50 = 3300 nM T12119 CW21LJ 145964527 IC50 = 690 nM T12119 C5MJ1S 145964650 IC50 = 390 nM T12119 CONK20 145964797 IC50 = 1100 nM T12119 C3FDW1 145964875 IC50 = 13.2 nM T12119 C52JFC 145965453 IC50 = 0.1 nM T12119 CSK8Y1 145965486 IC50 = 88 nM T12119 C3RYM4 145965521 IC50 = 1800 nM T12119 C4P7UD 145965756 IC50 = 6 nM T12119 CR1U5T 145965937 IC50 = 1600 nM T12119 CL0UK1 145966092 IC50 = 15000 nM T12119 CF4KG8 145966356 IC50 = 140 nM T12119 CIT81A 145966383 IC50 = 510 nM T12119 CYB3D7 145967129 IC50 = 260 nM T12119 CHF13C 145967515 IC50 = 510 nM T12119 CS78CA 145967768 IC50 = 59 nM T12119 C3LPS8 145968406 IC50 = 0.5 nM T12119 CJC57R 145968919 IC50 = 430 nM T12119 CK7PN3 145969142 IC50 = 11 nM T12119 C4HF5M 145969366 IC50 = 5 nM T12119 C5H0PQ 145969371 IC50 = 25000 nM T12119 C05NCW 145969596 IC50 = 6300 nM T12119 C94URS 145969597 IC50 = 2 nM T12119 CPXV56 145971430 IC50 = 170 nM T12119 CL9IA8 145971829 IC50 = 2340 nM T12119 C8BTO9 145971918 IC50 = 1.1 nM T12119 C4O5HA 145972742 IC50 = 4500 nM T12119 CD06JE 145972748 IC50 = 310 nM T12119 CS2T8H 145972807 IC50 = 4.8 nM T12119 COS4B9 145972887 IC50 = 1.1 nM T12119 C45IMD 145973060 IC50 = 100 nM T12119 CYP5U0 145973193 IC50 = 19.6 nM T12119 C5UE1S 145973817 IC50 = 0.5 nM T12119 C4XZ1W 145973987 IC50 = 48 nM T12119 C9H8ZW 145974032 IC50 = 29000 nM T12119 CC5U3D 145974386 IC50 = 0.12 nM T12119 CYX2V0 145974538 IC50 = 6.8 nM T12119 CS59YF 145974664 IC50 = 14 nM T12119 C1EH5C 145975024 IC50 = 1800 nM T12119 CT6Q3V 145975287 IC50 = 920 nM T12119 CHD75R 145975458 IC50 = 0.7 nM T12119 CP92XY 145975640 IC50 = 770 nM T12119 C12LRO 145975856 IC50 = 1700 nM T12119 CC49BG 145975892 IC50 = 170 nM T12119 CV0S3R 145976338 IC50 = 1500 nM T12119 C59HVM 145977053 IC50 = 1500 nM T12119 CMX4B2 145977179 IC50 = 2500 nM T12119 C7KZO2 145977238 IC50 = 94 nM T12119 CC1EP9 145977316 IC50 = 70 nM T12119 CT23DE 145977330 IC50 = 200 nM T12119 CH4IL5 145977429 IC50 = 350 nM T12119 CN9Q2I 145977501 IC50 = 28 nM T12119 CUV49K 145977796 IC50 = 34 nM T12119 C6XLF7 145978219 IC50 = 1150 nM T12119 C07URC 145978291 IC50 = 9700 nM T12119 C4O0KS 145978491 IC50 = 200 nM T12119 C3QB6J 145978986 IC50 = 350 nM T12119 CBR59Z 145979069 IC50 = 160 nM T12119 CUXB52 145979881 IC50 = 800 nM T12119 C87TKG 145980518 IC50 = 110 nM T12119 C7XK3P 145981121 IC50 = 1220 nM T12119 C96RZD 145981322 IC50 = 10 nM T12119 C8RA5D 145981858 IC50 = 640 nM T12119 CK5SA9 145982034 IC50 = 0.5 nM T12119 CZN0U6 145982478 IC50 = 5100 nM T12119 C1YW4D 145982684 IC50 = 370 nM T12119 CBK7Z6 145986895 IC50 = 210 nM T12119 C4GA2N 145987154 IC50 = 1480 nM T12119 CNL1W0 145987554 IC50 = 460 nM T12119 CIF5A3 145987886 IC50 = 14 nM T12119 C8Q2EG 145988110 IC50 = 1800 nM T12119 CP21ZQ 145988400 IC50 = 350 nM T12119 C8G1TO 145988654 IC50 = 60 nM T12119 CP45ZX 145988718 IC50 = 580 nM T12119 CW49OS 145990179 IC50 = 150 nM T12119 C6U7LS 145990658 IC50 = 420 nM T12119 C42YMJ 145990677 IC50 = 250 nM T12119 CHZB80 145990751 IC50 = 950 nM T12119 CGP61R 145991617 IC50 = 210 nM T12119 C0E2AZ 145991842 IC50 = 200 nM T12119 CMP27V 145992366 IC50 = 350 nM T12119 CQY2K6 145992782 IC50 = 720 nM T12119 CF48TY 145992899 IC50 < 10000 nM T12119 CDG51F 145993858 IC50 = 340 nM T12119 CN86HU 145994027 IC50 = 310 nM T12119 CW3B0G 145994131 IC50 = 620 nM T12119 C6DRM1 147449714 IC50 = 1100 nM T12119 C12NUF 149464333 IC50 = 1500 nM T12119 CI5NJ9 155510562 Ki = 0.68 nM T12119 CQKM15 155510624 IC50 = 1800 nM T12119 CM39UR 155510874 IC50 = 123 nM T12119 C6Q2PL 155511032 IC50 = 37 nM T12119 CNJ74U 155511848 IC50 = 314 nM T12119 C3LFE7 155512957 IC50 = 383 nM T12119 CXAL69 155513487 IC50 > 30000 nM T12119 CU63BY 155514109 IC50 = 642 nM T12119 C4MX5F 155516505 IC50 = 570 nM T12119 C30OPH 155516574 IC50 = 360 nM T12119 C8DA2L 155516676 IC50 = 660 nM T12119 CKM12Q 155517066 Ki = 1.7 nM T12119 C4W6SR 155517129 IC50 = 290 nM T12119 CY5UE9 155517299 IC50 = 2540 nM T12119 C8R0GW 155518443 Ki = 0.93 nM T12119 C03QEN 155519060 IC50 = 79 nM T12119 CM96HX 155520010 IC50 = 13 nM T12119 C64CPB 155520812 IC50 = 440 nM T12119 CAG7J0 155521246 IC50 = 20000 nM T12119 C76JKY 155521282 IC50 = 1550 nM T12119 C3A1YG 155522007 IC50 = 52 nM T12119 C9YAD2 155522119 Ki = 2.9 nM T12119 C26JPN 155523322 IC50 = 63 nM T12119 CV57GR 155523390 IC50 = 38 nM T12119 C65NKP 155524061 IC50 = 170 nM T12119 CO56NT 155524941 Ki = 3.9 nM T12119 CTM01D 155525057 IC50 = 85 nM T12119 C21CEX 155526133 IC50 = 280 nM T12119 C9RQ1Z 155526268 IC50 = 42 nM T12119 CZX19C 155526353 IC50 = 270 nM T12119 CF12TX 155527767 IC50 = 43 nM T12119 CRE0O6 155528016 IC50 = 3040 nM T12119 C1I0MA 155528300 IC50 = 1500 nM T12119 CU4VT6 155529277 Ki = 0.32 nM T12119 C5P0YG 155529298 IC50 = 850 nM T12119 CQOZ51 155529310 Ki = 18 nM T12119 C9U8FN 155529326 IC50 = 200 nM T12119 C6DJ5W 155530233 IC50 = 1400 nM T12119 C4PR0S 155530319 IC50 > 30000 nM T12119 CQ15KS 155530714 IC50 = 72 nM T12119 CU6NS9 155531543 IC50 = 720 nM T12119 CGO81N 155532622 IC50 = 1620 nM T12119 CZ3F2O 155533245 IC50 > 30000 nM T12119 CQE8Y5 155534372 IC50 = 1240 nM T12119 CXA95Z 155535618 IC50 = 509 nM T12119 CYC8R1 155535685 IC50 = 45 nM T12119 C87RFO 155536189 IC50 = 194 nM T12119 CO9HF7 155536553 Ki = 0.76 nM T12119 CO71LS 155536843 IC50 = 350 nM T12119 CMA9Q2 155537052 IC50 = 46 nM T12119 CA53FQ 155537146 IC50 = 890 nM T12119 C3KCV2 155537263 Ki = 1.5 nM T12119 CSDO95 155538523 IC50 > 30000 nM T12119 C64QKD 155538732 IC50 = 14 nM T12119 CW1D7Y 155538889 IC50 = 62 nM T12119 CRQW26 155539819 IC50 = 1100 nM T12119 CH63BD 155540878 IC50 = 260 nM T12119 CQO68V 155541113 IC50 = 388 nM T12119 C51KNE 155543494 IC50 = 1200 nM T12119 CEL05R 155543885 IC50 = 460 nM T12119 CQ7W0S 155544240 IC50 > 30000 nM T12119 C74VOU 155544985 IC50 = 2000 nM T12119 CXHL65 155545824 Ki = 1 nM T12119 CZ47YD 155545889 IC50 = 160 nM T12119 CEPJ20 155545982 IC50 = 10600 nM T12119 CY0AM8 155547012 IC50 > 42000 nM T12119 CINZ05 155547490 IC50 > 42000 nM T12119 CZCB86 155547694 IC50 = 7820 nM T12119 CPD1B3 155547824 IC50 = 510 nM T12119 CI74WT 155548729 IC50 = 30 nM T12119 CI94QY 155550095 IC50 = 140 nM T12119 C4DF0X 155550384 Ki = 2.9 nM T12119 C1GBV3 155551722 IC50 > 30000 nM T12119 CWFH54 155552017 IC50 = 85 nM T12119 CDIZ34 155552658 Ki = 0.51 nM T12119 C1WTQ7 155553777 IC50 = 635 nM T12119 CAV3Q9 155553847 IC50 > 30000 nM T12119 CT4X3F 155554021 IC50 = 1100 nM T12119 CMI0U2 155554255 IC50 = 3020 nM T12119 C34SWX 155554756 Ki = 1.3 nM T12119 CGE76T 155555738 IC50 > 30000 nM T12119 CJX1Q7 155557620 IC50 = 200 nM T12119 C0AH6G 155557721 IC50 = 1800 nM T12119 CK89PG 155557967 IC50 = 116 nM T12119 C0T6WM 155558045 IC50 = 10700 nM T12119 CU4FQ3 155558358 IC50 > 30000 nM T12119 C71TVP 155559515 IC50 = 680 nM T12119 CZ0VL5 155559622 IC50 = 1200 nM T12119 CY06UB 155561401 IC50 = 70 nM T12119 CL96XW 155562578 IC50 > 30000 nM T12119 CPL2D9 155562982 IC50 = 150 nM T12119 CSDR68 155563772 IC50 = 48 nM T12119 CNLE43 155564167 IC50 > 42000 nM T12119 CJL8Y5 155565696 IC50 = 280 nM T12119 C2EKM7 155566527 IC50 = 104 nM T12119 CZ9OW6 155567417 IC50 > 30000 nM T12119 CG97KZ 155568180 IC50 = 550 nM T12119 D00TGC 56951318 IC50 = 80 nM T12119 D02HMZ 11427214 IC50 = 2160 nM T12119 D02PZJ 11324184 IC50 = 1940 nM T12119 D0F5MZ 11460438 IC50 = 5310 nM T12119 D0FF6S 16038374 IC50 = 6740 nM T12119 D0M1OU 11998198 IC50 = 3 nM T12119 D0P8TL 56947150 IC50 = 702 nM T86503 C16CXQ 10033400 Ki = 240 nM T86503 CBUF92 11228390 Ki = 0.4 nM T86503 CJ73BT 45486346 Ki = 42 nM T86503 C9ETC4 45486354 Ki = 67 nM T86503 CVPG40 45486356 Ki = 3 nM T86503 CSQ2K4 45486357 Ki = 2.4 nM T86503 C6TO1L 71450124 Ki = 70 nM T86503 C8F5YQ 71451941 Ki > 1000 nM T86503 CGD6J4 71451942 Ki = 18 nM T86503 CY86ZW 71453763 Ki = 1600 nM T86503 C5I3EB 71453792 Ki = 23 nM T86503 CT51YJ 71453793 Ki = 1.1 nM T86503 C7WM6Z 71455497 Ki = 20 nM T86503 C35YRK 71457282 Ki = 1380 nM T86503 C2YEU4 71457318 Ki = 24 nM T86503 CB9MG1 71459125 Ki = 0.34 nM T86503 C0N8UR 71460934 Ki = 1.3 nM T86503 CDLP98 71460935 Ki = 2 nM T86503 CIS3R0 71460936 Ki = 300 nM T86503 CK1X0W 71462644 Ki = 7 nM T86503 CGR35S 71462645 Ki = 1600 nM T86503 CQNG13 71608634 Ki = 4.9 nM T86503 C4APW2 75593416 Ki = 14 nM T86503 CJ2W9V 75593418 Ki = 5.3 nM T86503 C29QOJ 76310654 Ki = 6260 nM T86503 CAT6S5 76310655 Ki = 14000 nM T86503 CG87ZE 76310656 Ki = 14000 nM T86503 CV8Z5G 76314290 Ki = 25 nM T86503 CGB4J9 76317836 Ki = 21 nM T86503 C7G4XB 76317837 Ki = 27 nM T86503 CFXK67 76317855 Ki = 57 nM T86503 CH3N0A 76321557 Ki = 385 nM T86503 CF78UP 76321572 Ki = 60 nM T86503 CMYK97 76325157 Ki = 39 nM T86503 CZ62KS 76328735 Ki = 170 nM T86503 C4LG2O 76328736 Ki = 350 nM T86503 CIY15Q 76332398 Ki = 500 nM T86503 CL2ZX3 76332418 Ki = 700 nM T86503 CX2VL4 76336024 Ki = 400 nM T86503 CGZN04 76336044 Ki = 960 nM T86503 C0ET8W 137630787 Ki = 3.6 nM T86503 CC3V7S 137631353 Ki = 4 nM T86503 C2JV6R 137631479 Ki = 0.3 nM T86503 C53MJF 137631755 Ki = 3 nM T86503 CN26ME 137631991 Ki = 14 nM T86503 CUOC87 137632800 Ki = 2.5 nM T86503 C5VFZ9 137633317 Ki = 6 nM T86503 C73DJB 137633620 Ki = 16 nM T86503 CBNJ52 137633770 Ki = 4.8 nM T86503 CRN21S 137633930 Ki = 60 nM T86503 CP8DN5 137634404 Ki = 2 nM T86503 CAIC85 137634503 Ki = 4 nM T86503 C0T3NR 137635077 Ki = 4 nM T86503 C9MUE6 137636542 Ki = 2.8 nM T86503 CG95RB 137636600 Ki = 5 nM T86503 C4GHK8 137636619 Ki = 5 nM T86503 CG5Q8T 137636730 Ki = 1 nM T86503 CH8AU1 137636950 Ki = 18 nM T86503 CDVJ93 137637528 Ki = 39 nM T86503 C5DX1A 137637600 Ki = 3 nM T86503 CDY46K 137637620 Ki = 400 nM T86503 C87STU 137638937 Ki = 10 nM T86503 C5L0NC 137639050 Ki = 6 nM T86503 CBH65X 137639397 Ki = 18 nM T86503 CN0FY7 137639688 Ki = 0.9 nM T86503 CJMG20 137640300 Ki = 8 nM T86503 CB2Z9N 137640311 Ki = 2.2 nM T86503 CERC30 137640559 Ki = 1.3 nM T86503 C35AYG 137641095 Ki = 5 nM T86503 CUM15D 137641134 Ki = 140 nM T86503 CQ76RK 137641874 Ki = 9 nM T86503 CO3S8F 137641997 Ki = 6 nM T86503 CMA50S 137642172 Ki = 0.4 nM T86503 C5AM0F 137642389 Ki = 4.1 nM T86503 CNC1O3 137642533 Ki = 44 nM T86503 CA5PJ2 137642642 Ki = 2 nM T86503 CX53VG 137642650 Ki = 46 nM T86503 CHI60U 137642806 Ki = 0.2 nM T86503 C7W9US 137643496 Ki = 3 nM T86503 C7PR9K 137644391 Ki = 2 nM T86503 C98VOE 137645351 Ki = 1 nM T86503 C0NWD3 137645581 Ki = 36 nM T86503 CQ6SI9 137645677 Ki = 8 nM T86503 CJT5C4 137646929 Ki = 6 nM T86503 C8WED4 137647032 Ki = 0.4 nM T86503 C76BDY 137647768 Ki = 2.8 nM T86503 CD3CZ6 137647834 Ki = 3 nM T86503 C64QUK 137648887 Ki = 80 nM T86503 CBP37G 137649385 Ki = 8 nM T86503 C2N9LT 137650514 Ki = 4 nM T86503 COR8J3 137652054 Ki = 8 nM T86503 CJX57S 137652059 Ki = 2.1 nM T86503 CVC56D 137652453 Ki = 30 nM T86503 CUP70F 137652558 Ki = 3.7 nM T86503 CJVG81 137652912 Ki = 51 nM T86503 CPO80U 137653066 Ki = 5 nM T86503 CN5VC7 137653379 Ki = 9.8 nM T86503 C34XTZ 137653755 Ki = 2 nM T86503 CUHM58 137653788 Ki = 1.5 nM T86503 C4B8DK 137654788 Ki = 9 nM T86503 C4XTJ7 137655341 Ki = 4 nM T86503 C7W1GU 137655527 Ki = 2 nM T86503 CBRA14 137655621 Ki = 3 nM T86503 CI78BN 137656445 Ki = 2 nM T86503 CD9N0S 137656589 Ki = 12 nM T86503 CV7T5U 137656624 Ki = 21 nM T86503 CI3A4J 137657514 Ki = 0.6 nM T86503 CO09SX 137658594 Ki = 1.7 nM T86503 CZY51S 137659359 Ki = 0.5 nM T86503 C8J2FS 137659865 Ki = 4 nM T86503 CXYA13 137660373 Ki = 4 nM T86503 C37WVK 137660935 Ki = 28 nM T86503 CGBP12 137661234 Ki = 2 nM T86503 CSI79D 137661408 Ki = 6.2 nM T86503 CV3NU9 137661582 Ki = 1.8 nM T86503 CDP9F6 145979561 Ki = 17 nM T86503 C0FVL7 145980400 Ki = 700 nM T86503 C7U6AC 145980921 Ki = 14 nM T86503 C1PY3D 145982564 Ki = 150 nM T86503 C0F2HS 145982570 Ki = 64 nM T86503 C9BAM3 145982642 Ki = 160 nM T86503 CO1L7J 145982755 Ki = 58 nM T86503 CH49CQ 145982874 Ki = 68 nM T86503 CL4F2V 145983062 Ki = 30 nM T86503 C8P4IY 145983083 Ki = 70 nM T86503 CD4V6Y 145983456 Ki = 22 nM T86503 C0VPE7 145983531 Ki = 250 nM T86503 CMN3C0 145983800 Ki = 37 nM T86503 CKY29N 145984016 Ki = 11 nM T86503 C71KAW 145984052 Ki = 33 nM T86503 C7Y5TR 145984180 Ki = 64 nM T86503 CI2E5Y 145984243 Ki = 20 nM T86503 CP4M8O 145984298 Ki = 32 nM T86503 CR0E5D 145984449 Ki = 28 nM T86503 CBK18Y 145984711 Ki = 29 nM T86503 C9W1TO 145984728 Ki = 41 nM T86503 CZ9MK3 145984956 Ki = 170 nM T86503 C6VYO5 145985131 Ki = 44 nM T86503 C0DJ8X 145985285 Ki = 32 nM T86503 CME81P 145985674 Ki = 248 nM T86503 CMT30D 145985833 Ki = 29 nM T86503 CN96XK 145985989 Ki = 38 nM T86503 C6UA9H 145986239 Ki = 43 nM T86503 CG7LW4 145987687 Ki = 13 nM T86503 C3C2LW 145989654 Ki = 500 nM T86503 C4IW1B 145989737 Ki = 53 nM T86503 C4ACG5 145990382 Ki = 240 nM T86503 CZJY41 145990864 Ki = 2.6 nM T86503 CB9FH7 145992096 Ki = 190 nM T86503 C9KC4Q 145993075 Ki = 32 nM T86503 D0A6FZ 75593419 Ki = 3.1 nM T86503 D0Y9PH 45486355 Ki = 0.6 nM T54771 D01TNW 9887712 IC50 = 3.2 nM T54771 D04DXA 46908929 IC50 = 8444 nM T54771 D06ALD 11949646 EC50 = 8300 nM T54771 D08DFX 24812758 IC50 = 684 nM T54771 D0Q3VE 44814423 IC50 = 392 nM T54771 D07FBM 10453870 EC50 = 1900 nM T54771 D0IJ0U 11988953 IC50 = 3990 nM T54771 D0OR3G 25195624 IC50 = 2.3 nM T54771 D0U7IL 24831714 IC50 = 34.6 nM T54771 CZN6S9 743974 IC50 > 39810.72 nM T54771 C7BS0Y 1226045 IC50 = 7900 nM T54771 C6D3EB 2822337 IC50 = 7000 nM T54771 CXWS61 3086055 IC50 = 13300 nM T54771 C1R8VD 6474295 IC50 = 25400 nM T54771 CZI0R5 6918439 Ki = 50 nM T54771 CIX6M9 9800802 IC50 = 540 nM T54771 CL1I4S 9953041 IC50 = 442 nM T54771 C38QWM 9956975 IC50 = 60 nM T54771 CD81IB 10009210 IC50 = 11 nM T54771 CC8KZ7 10073130 IC50 = 446 nM T54771 CQW18C 10133993 IC50 = 9300 nM T54771 CL8U9W 10301121 IC50 = 37 nM T54771 C8WUG3 10388250 IC50 = 392 nM T54771 C9G0BJ 10431578 IC50 = 320 nM T54771 CIV50R 10434911 IC50 = 931 nM T54771 CEO3K9 10453180 IC50 = 422 nM T54771 C4XW1Y 10778685 IC50 = 25600 nM T54771 CDG74B 10806690 IC50 = 34600 nM T54771 C30MWO 10812923 IC50 = 10400 nM T54771 C9H8PW 11155568 IC50 = 2240 nM T54771 CPJ58S 11166239 IC50 = 3200 nM T54771 C8ZN5I 11177436 IC50 = 2140 nM T54771 CHV85J 11177940 IC50 = 2890 nM T54771 CP93BY 11282187 IC50 = 3050 nM T54771 C56VGN 11305464 IC50 = 1100 nM T54771 CTA3F7 11383983 IC50 = 4390 nM T54771 CG7A2S 11385553 IC50 = 3610 nM T54771 CLG02Z 11397072 IC50 = 1970 nM T54771 COPU18 11419680 IC50 = 198 nM T54771 CQ98CT 11441784 IC50 = 611 nM T54771 CXD46E 11442119 IC50 = 1190 nM T54771 CG6W5A 11452732 IC50 = 1510 nM T54771 C9GFV6 11502260 IC50 = 31000 nM T54771 C0H4YI 11509368 IC50 = 3500 nM T54771 C0IC5X 11509608 IC50 > 100000 nM T54771 CE76UG 11510297 IC50 = 8600 nM T54771 C67HDU 11516541 IC50 = 5600 nM T54771 CGY18M 11517178 IC50 = 57000 nM T54771 C2D8PW 11524511 IC50 = 4500 nM T54771 CKI73F 11530288 IC50 = 13000 nM T54771 CXD1G4 11531141 IC50 = 7800 nM T54771 C9IJ0T 11546717 IC50 = 718 nM T54771 CH01CX 11552436 IC50 = 3300 nM T54771 CG0AL2 11552441 IC50 = 25000 nM T54771 CN4MY1 11553111 IC50 > 100000 nM T54771 C86MYU 11559484 IC50 = 33000 nM T54771 CTR8Z2 11560149 IC50 = 41000 nM T54771 CZ79RA 11566856 IC50 = 27000 nM T54771 C2Q9YI 11596174 IC50 = 73000 nM T54771 C3I5OZ 11631863 IC50 = 19000 nM T54771 C0U9BG 11639042 IC50 = 6700 nM T54771 C8GS9Z 11646163 IC50 = 48000 nM T54771 C3CY4U 11654569 IC50 = 210 nM T54771 C4D1CR 11660874 IC50 = 22000 nM T54771 CW54RB 11675148 IC50 = 4800 nM T54771 CFAP86 11682042 IC50 = 38000 nM T54771 C7Y0MN 11689581 IC50 = 510 nM T54771 CKFJ21 11703862 IC50 = 720 nM T54771 CDTY94 11704386 IC50 > 100000 nM T54771 CYK57O 11718001 IC50 > 100000 nM T54771 CQM7K2 11718002 IC50 = 20000 nM T54771 C08ZYC 11744475 IC50 = 831 nM T54771 C2Y5LI 11751069 IC50 = 145 nM T54771 CTF76L 11758523 IC50 = 50 nM T54771 C7HZ5B 11949311 IC50 = 0.16 nM T54771 C89EKZ 11949687 IC50 = 8300 nM T54771 CIFG87 11989083 IC50 = 4040 nM T54771 C0VF4G 12044949 IC50 = 33900 nM T54771 C5FC3A 13990811 IC50 = 50900 nM T54771 CMX78G 15979165 IC50 = 9.6 nM T54771 CYT6R3 21722188 IC50 = 19000 nM T54771 C09GWO 23581834 IC50 = 600 nM T54771 C7FZW6 23581843 IC50 = 28 nM T54771 C2L8YJ 23725183 EC50 = 27 nM T54771 CF1B5J 24759836 IC50 = 230 nM T54771 C3AE6U 24764501 IC50 = 1900 nM T54771 CSTE65 24768285 EC50 > 8000 nM T54771 CB78ZL 24822185 IC50 = 25 nM T54771 CE48BP 24851760 IC50 = 764 nM T54771 C15MTU 24851762 IC50 = 65 nM T54771 C4MH7I 24851868 IC50 = 175 nM T54771 C4NLZ8 24948046 IC50 = 4200 nM T54771 CWGV89 24989734 IC50 = 65 nM T54771 C1VP4M 24989735 IC50 = 32 nM T54771 COH9F6 25168565 IC50 = 91000 nM T54771 C9PYQ3 25168566 IC50 > 10000 nM T54771 CA3F4Z 25168568 IC50 = 60000 nM T54771 C2SLA9 25168702 IC50 > 1000 nM T54771 CN7TU2 25168703 IC50 > 10000 nM T54771 C0STB7 25168704 IC50 > 10000 nM T54771 CZ3N7V 25168707 IC50 = 31000 nM T54771 CTX09K 25168849 IC50 = 103000 nM T54771 CM20EO 25168980 IC50 > 20000 nM T54771 CT6J9S 25169379 IC50 > 5000 nM T54771 C96QDH 25169515 IC50 = 140000 nM T54771 CVWR84 25174140 IC50 = 6 nM T54771 CE2R4Z 25197075 IC50 = 3 nM T54771 C9E3KT 25197183 IC50 = 10 nM T54771 CJBE59 25197291 IC50 = 8 nM T54771 CEV78S 25197294 IC50 = 9.6 nM T54771 CCW2Z3 25197296 IC50 = 4 nM T54771 C76CAY 25224975 IC50 = 750 nM T54771 CV36FX 29977194 Ki = 560 nM T54771 C7E3IS 44236835 IC50 = 1.8 nM T54771 CE7A4F 44236838 IC50 = 10 nM T54771 CI40RV 44236839 IC50 = 3 nM T54771 CU2PY7 44291236 Ki = 2600 nM T54771 C59ETX 44394297 Ki = 8590 nM T54771 CJA5P8 44394328 Ki = 8390 nM T54771 CWF4S2 44394360 Ki = 6280 nM T54771 CKQ8C4 44394366 Ki = 16100 nM T54771 COEQ58 44394379 Ki = 1320 nM T54771 C1LR5Q 44394382 Ki = 4780 nM T54771 CM34LN 44394389 Ki = 4380 nM T54771 CAX9I5 44394395 Ki = 1380 nM T54771 C4FAS7 44394396 Ki = 3690 nM T54771 CHD62C 44394401 Ki = 33100 nM T54771 CE95IS 44394404 Ki = 1570 nM T54771 CRT40X 44394412 Ki = 4640 nM T54771 CH4YD2 44394431 Ki = 1460 nM T54771 C0GB3P 44394436 Ki = 3750 nM T54771 CA9IK4 44394445 Ki = 1080 nM T54771 CYJ6Q1 44394447 Ki > 45000 nM T54771 C0S2TF 44394455 Ki = 6500 nM T54771 C20IMQ 44394486 Ki > 45000 nM T54771 CV9M5H 44394509 Ki = 13520 nM T54771 CN7A4F 44394518 Ki > 45000 nM T54771 CSRJ24 44394527 Ki = 16150 nM T54771 CG6MK7 44394566 Ki = 9890 nM T54771 CGFX45 44580555 IC50 = 9.4 nM T54771 CVYJ93 44626350 IC50 = 620 nM T54771 C3VT8W 44626351 IC50 = 10000 nM T54771 CH2SF6 45101268 IC50 = 3060 nM T54771 CVEI19 45101270 IC50 = 3988 nM T54771 C98KYC 45101303 IC50 > 10000 nM T54771 CDJ8G6 45101306 IC50 > 10000 nM T54771 CU31BJ 45101308 IC50 = 820 nM T54771 C9QN4L 45101346 IC50 = 7000 nM T54771 CN7SY1 45101347 IC50 = 900 nM T54771 CKY7J1 45101349 IC50 = 3170 nM T54771 CX5B3E 45488013 IC50 = 700 nM T54771 CK3W2T 45488018 IC50 = 2700 nM T54771 CX6HS7 45488023 IC50 = 200 nM T54771 CG1X9S 45488025 IC50 = 2500 nM T54771 CLOC07 45488026 IC50 = 10500 nM T54771 CD1R8X 45488027 IC50 = 10000 nM T54771 C4QBL8 45488028 IC50 = 14000 nM T54771 CKNR92 45488030 IC50 = 1000 nM T54771 CE35BT 45488037 IC50 = 3500 nM T54771 CR1OQ2 45488039 IC50 = 1000 nM T54771 C7E6TD 45488040 IC50 > 100000 nM T54771 C0DY9S 45488049 IC50 = 10000 nM T54771 C1XO0E 45488050 IC50 = 43000 nM T54771 C1QI8N 45488053 IC50 = 1000 nM T54771 CGJ30Y 45488055 IC50 = 1600 nM T54771 C6SY0U 45488063 IC50 = 18745 nM T54771 CB6HD1 45488064 IC50 = 10000 nM T54771 CF4O8U 45488065 IC50 = 6000 nM T54771 CFH24W 45488067 IC50 = 9700 nM T54771 C1VI8W 45488068 IC50 = 3100 nM T54771 C2L4DC 45488083 IC50 = 1500 nM T54771 CXQ43I 45488084 IC50 = 1000 nM T54771 CI2QE1 45488087 IC50 = 5300 nM T54771 CPCY36 46195348 IC50 = 5040 nM T54771 CPI96D 46201936 IC50 = 5600 nM T54771 CPI7Y6 46204509 IC50 = 26100 nM T54771 C8VRT9 46204510 IC50 = 14600 nM T54771 CA2T3C 46204511 IC50 = 565 nM T54771 C2ROV8 46204818 IC50 = 7960 nM T54771 C16TNB 46204819 IC50 = 671 nM T54771 CY2R7X 46204820 IC50 = 1210 nM T54771 CYH76W 46204821 IC50 = 100000 nM T54771 CIR8F2 46204822 IC50 = 4270 nM T54771 C0YOD9 46204823 IC50 = 260 nM T54771 CXD41T 46205138 IC50 = 209 nM T54771 CNBV15 46205139 IC50 = 602 nM T54771 CT2B4U 46205140 IC50 = 8160 nM T54771 C48RLS 46205141 IC50 = 35600 nM T54771 CD25IE 46205142 IC50 = 391 nM T54771 C9BAU2 46205143 IC50 = 2830 nM T54771 CXGD79 46205461 IC50 = 17300 nM T54771 CV1JB3 46205462 IC50 = 3340 nM T54771 C87XZS 46206829 IC50 = 1540 nM T54771 C3NO5G 46206830 IC50 = 1500 nM T54771 CU0GS3 46206831 IC50 > 10000 nM T54771 CR6C8O 46206832 IC50 > 10000 nM T54771 CK28MY 46206833 IC50 > 9600 nM T54771 CKV8G1 46210599 IC50 = 27000 nM T54771 C1C8DJ 46210600 IC50 = 37000 nM T54771 C4JEC9 46229153 IC50 = 17000 nM T54771 C01HGP 46229154 IC50 = 50000 nM T54771 CN1B9F 46229155 IC50 = 5000 nM T54771 C1J7NT 46229156 IC50 = 4000 nM T54771 COF9A7 46229157 IC50 = 5000 nM T54771 CEI97D 46229158 IC50 > 100000 nM T54771 C0NE3T 46229159 IC50 = 97000 nM T54771 CPO40S 46229160 IC50 > 100000 nM T54771 CJ61SL 46861619 IC50 = 35 nM T54771 C4IP5Z 46865788 IC50 = 190 nM T54771 CG50FN 46865896 IC50 = 370 nM T54771 CQ04HT 46881709 IC50 = 73 nM T54771 C4EQH7 46881761 IC50 = 6800 nM T54771 CI9VO5 46881762 IC50 = 1100 nM T54771 C39CJH 46897476 IC50 = 35 nM T54771 CG3IL5 46897478 IC50 = 46 nM T54771 C6Q0NU 46897565 IC50 = 54 nM T54771 C1CZ4A 46897566 IC50 = 29 nM T54771 CRF28B 46897567 IC50 = 42 nM T54771 C5UWM8 46897656 IC50 = 30 nM T54771 C7OW4N 46897658 IC50 = 27 nM T54771 CMGI18 46906366 IC50 > 2000 nM T54771 CF2K6T 46906391 IC50 = 134000 nM T54771 C6JKR2 46906469 IC50 > 2000 nM T54771 CRV61E 50925634 EC50 = 208.6 nM T54771 C30UZQ 50942027 IC50 = 9900 nM T54771 C6SP8V 50992818 EC50 = 229.5 nM T54771 C7Y2IX 50992875 EC50 = 233.9 nM T54771 CGN81J 50992876 EC50 = 327.3 nM T54771 CD3N4X 50993708 EC50 = 628.8 nM T54771 C2XLV3 50993712 EC50 = 305.9 nM T54771 C4YF1K 50993787 EC50 = 461.6 nM T54771 C9VI3M 52918252 IC50 = 9140 nM T54771 C1AE6L 52918253 IC50 = 6290 nM T54771 C3X1MP 52944051 IC50 = 910 nM T54771 CNI2X3 52952611 IC50 > 10000 nM T54771 CK7EW5 52952725 IC50 = 546 nM T54771 CH03OA 52952726 IC50 > 10000 nM T54771 CMW1K2 53363122 IC50 = 4.4 nM T54771 CFJ5G8 53389526 IC50 = 30000 nM T54771 CVR7K0 53467552 IC50 > 90000 nM T54771 CVL86S 53467553 IC50 > 90000 nM T54771 C2ED6O 53467554 IC50 > 90000 nM T54771 CW40YV 53467555 IC50 > 90000 nM T54771 CX7P2D 53467556 IC50 > 90000 nM T54771 C5YX0V 53467759 IC50 > 90000 nM T54771 C8CLN9 53467761 IC50 > 90000 nM T54771 C7Q6AJ 53467762 IC50 > 90000 nM T54771 C92DHW 53467763 IC50 > 90000 nM T54771 C6O3NH 53467764 IC50 > 90000 nM T54771 C0T5VA 53467975 IC50 > 90000 nM T54771 C78TRY 53468202 IC50 = 35308 nM T54771 C2N8AH 53468203 IC50 = 83060 nM T54771 C7VQG5 53468204 IC50 = 90000 nM T54771 C2XHO3 53468206 IC50 = 17500 nM T54771 C31UEL 53468414 IC50 = 6252 nM T54771 C1NJ5P 54579981 IC50 = 7340 nM T54771 CL4K3S 54579982 IC50 = 7280 nM T54771 C7A5FM 54580749 IC50 = 506 nM T54771 CAL4P2 54580976 IC50 = 13600 nM T54771 CZ0MV1 54580977 IC50 = 13800 nM T54771 CLJ76E 54581991 IC50 = 3750 nM T54771 CYW6B8 54581992 IC50 = 6640 nM T54771 C0QA6R 54582021 IC50 = 25000 nM T54771 C1N0KC 54582874 IC50 = 30000 nM T54771 CP8L4K 54582928 IC50 = 4750 nM T54771 COS5F2 54582929 IC50 = 5610 nM T54771 CO82HW 54582930 IC50 = 7340 nM T54771 CJ6WB3 54582969 IC50 = 46000 nM T54771 C46EPV 54582970 IC50 = 9880 nM T54771 C5EPU2 54583960 IC50 = 6900 nM T54771 CV2R1U 54584874 IC50 = 3470 nM T54771 CLH1P6 54584875 IC50 = 7130 nM T54771 C7KRD4 54584876 IC50 = 2530 nM T54771 C5W0CS 54585841 IC50 = 2000 nM T54771 CNIF43 54585871 IC50 = 11800 nM T54771 CW6H2Y 54586611 IC50 = 958 nM T54771 CLM0E5 54586807 IC50 = 5320 nM T54771 C0A1GD 54586808 IC50 = 3290 nM T54771 CMA48J 56673660 IC50 = 428 nM T54771 CTL9A8 56676982 IC50 = 93 nM T54771 C34PBD 56942482 IC50 = 38 nM T54771 C7M0QO 57556376 IC50 = 6281 nM T54771 CPS65X 57556380 IC50 = 18697 nM T54771 C7E8MR 57556391 IC50 = 12335 nM T54771 CJ59CN 57556398 IC50 = 5902 nM T54771 CP82CI 57556406 IC50 = 13137 nM T54771 CIL8S9 57556409 IC50 = 24146 nM T54771 CUL1T8 57556416 IC50 = 126 nM T54771 C9OW3L 57556425 IC50 = 8482 nM T54771 CZ5B2H 57556428 IC50 = 28918 nM T54771 CL52JF 57556430 IC50 = 4987 nM T54771 CF70BA 57556431 IC50 = 81487 nM T54771 CO01YH 57556433 IC50 = 3086 nM T54771 C5IY8V 57802355 IC50 = 689 nM T54771 CZ9N7D 57802433 IC50 = 94 nM T54771 CTA1V4 58178431 IC50 = 9900 nM T54771 C2VP8M 58186566 IC50 = 1956 nM T54771 CQ1RO6 58239014 IC50 = 162 nM T54771 C6I4LS 58507570 IC50 = 388 nM T54771 CH4JP5 60134927 IC50 = 5314 nM T54771 C4AHP2 66691967 IC50 = 9600 nM T54771 CPB6R3 67196949 IC50 = 22 nM T54771 CHS7E9 67304774 IC50 = 51 nM T54771 CAM0S1 68535905 IC50 = 23 nM T54771 C6XLO5 68537281 IC50 = 70 nM T54771 CIOM04 68538795 IC50 = 15 nM T54771 CU2YH4 68538810 IC50 = 217 nM T54771 CY9W4S 68538834 IC50 = 772 nM T54771 CCP3K5 68540044 IC50 = 103 nM T54771 CHS98N 68540709 IC50 = 351 nM T54771 C02MEL 68542200 IC50 = 45 nM T54771 CS3BC9 69516549 IC50 = 9520 nM T54771 C0AS6H 69516684 IC50 = 306 nM T54771 CMB3H2 69516839 IC50 = 203 nM T54771 C29AIC 70681502 Ki > 1000000 nM T54771 C02YNI 70684428 EC50 = 23063 nM T54771 C3TL7D 70684429 EC50 = 282 nM T54771 CNM2G0 70686571 EC50 = 550 nM T54771 CL57CD 70687204 Ki = 14000 nM T54771 CDH53P 70688690 EC50 = 20937 nM T54771 C5SRW9 70690752 EC50 = 3208 nM T54771 CDR2S1 70692889 EC50 = 6427 nM T54771 COFW37 70692890 EC50 = 884 nM T54771 CLSI96 70692891 EC50 = 55 nM T54771 C47OBZ 70694930 EC50 = 9523 nM T54771 CX13VG 70696980 EC50 = 2491 nM T54771 C84IFU 70696981 EC50 = 4962 nM T54771 CC9AH0 71451518 IC50 = 2430 nM T54771 CV7Y2F 71453231 IC50 = 1720 nM T54771 CG9TO4 71453232 IC50 = 246 nM T54771 CB6Z5A 71453233 IC50 = 1330 nM T54771 C07IRW 71453345 IC50 = 675 nM T54771 C54QMZ 71454958 IC50 = 278 nM T54771 C3LBY4 71454959 IC50 = 871 nM T54771 C2BOR8 71454960 IC50 = 8930 nM T54771 CL5P0D 71454961 IC50 = 500 nM T54771 CZ6QB5 71454962 IC50 = 223 nM T54771 C61YGV 71455054 IC50 = 298 nM T54771 CA1SU7 71455055 IC50 = 738 nM T54771 CHGR43 71456753 IC50 = 1940 nM T54771 CDJ14N 71456754 IC50 = 4310 nM T54771 C6DRB5 71456755 IC50 = 207 nM T54771 CE6F9D 71457086 IC50 = 5132 nM T54771 C3DN7L 71458597 IC50 = 4310 nM T54771 CZWO59 71460439 IC50 = 1190 nM T54771 C69OZJ 71460532 IC50 = 7280 nM T54771 C7DMG8 71462125 IC50 = 1230 nM T54771 CMG4Y3 71462176 IC50 = 7170 nM T54771 CA6VK1 71462236 IC50 = 725 nM T54771 CT73OL 71524007 IC50 = 724 nM T54771 CM2LH3 71524008 IC50 = 1500 nM T54771 CH9SD8 71524009 IC50 = 1470 nM T54771 CX4Q0G 71524030 IC50 = 6170 nM T54771 C3E9IM 71524031 IC50 = 1990 nM T54771 C4IBY1 71524032 IC50 = 1030 nM T54771 COGI16 71524033 IC50 = 517 nM T54771 CH96ZJ 71524034 IC50 = 170 nM T54771 CEZ71U 71524035 IC50 = 12 nM T54771 CRC40T 71524036 IC50 = 10 nM T54771 CX8U3Q 71524037 IC50 = 25 nM T54771 CA1I2V 71524038 IC50 = 124 nM T54771 C70ITO 71603300 EC50 = 5424 nM T54771 CR8M7J 71604141 EC50 = 5933 nM T54771 CHS89O 71604142 EC50 = 12572 nM T54771 CBG14D 71604199 EC50 = 5390 nM T54771 CQ3T0D 71604202 EC50 = 18080 nM T54771 CL7R1O 71604268 EC50 = 4091 nM T54771 C4G6DV 71604269 EC50 = 4931 nM T54771 CZTA53 71604270 EC50 = 1412 nM T54771 CBX81V 71716041 Ki = 7700 nM T54771 C4QJ8B 71716042 Ki = 23100 nM T54771 CBG43K 71716640 Ki = 21600 nM T54771 CB8Y6D 71717244 Ki = 45000 nM T54771 CGPK29 71717245 Ki = 152000 nM T54771 CO1S6J 71717246 Ki = 116000 nM T54771 CI4CN3 71717852 Ki = 2800 nM T54771 C4CA8B 71718493 Ki = 7000 nM T54771 C9A6HG 71719073 Ki = 40000 nM T54771 CE1L9Z 71719074 Ki = 5300 nM T54771 CTU0E6 71719075 Ki = 3800 nM T54771 C38EAU 71719076 Ki = 94300 nM T54771 CH0DS6 71719684 Ki = 93100 nM T54771 CX0UM3 73346536 EC50 > 50000 nM T54771 CJ01LN 73348014 EC50 > 50000 nM T54771 C7GCY0 73348015 EC50 = 29000 nM T54771 CZ9AT7 73348017 EC50 > 50000 nM T54771 C2R0ZL 73349555 EC50 = 24000 nM T54771 CS97BC 73354077 EC50 > 50000 nM T54771 CKC2V7 73354078 EC50 > 50000 nM T54771 CYWE90 73354079 EC50 > 50000 nM T54771 CU0Z8P 73354081 EC50 > 50000 nM T54771 C9SZN5 73355608 EC50 = 47000 nM T54771 CW8XK6 73357149 EC50 > 50000 nM T54771 CNX4Y8 74538678 IC50 = 3.3 nM T54771 CUI04H 76070792 IC50 = 1.8 nM T54771 C65ICL 76070894 IC50 = 2.2 nM T54771 CC4U0L 76070897 IC50 = 2.3 nM T54771 C5TP1J 76070999 IC50 = 250 nM T54771 CCL50G 76071000 IC50 = 2.4 nM T54771 C60BEU 76071231 IC50 = 25.3 nM T54771 CMIF39 76310883 IC50 = 314.6 nM T54771 C5LZ9K 76310884 IC50 = 467.4 nM T54771 C21SOA 76314516 IC50 = 315.4 nM T54771 CE4MR2 76315186 IC50 = 10400 nM T54771 CPF3Q2 76318092 IC50 = 256.7 nM T54771 CX2H5F 76318093 IC50 = 628.5 nM T54771 CL2WO9 76321790 IC50 = 523.5 nM T54771 CE07JZ 76325427 IC50 = 621 nM T54771 CEKB95 76325428 IC50 = 392.2 nM T54771 C1ZP0V 76325429 IC50 = 434.1 nM T54771 C82SWJ 76325430 IC50 = 693.2 nM T54771 CF0R6P 76328964 IC50 = 527.5 nM T54771 C2T7KO 76332640 IC50 = 626.2 nM T54771 CXH87A 76336244 IC50 = 435.2 nM T54771 CLV1N4 76336245 IC50 = 466.8 nM T54771 C2G4YS 76336246 IC50 = 220 nM T54771 C4RY1I 86282875 IC50 = 1096 nM T54771 C2ZMG1 89630294 EC50 = 2027 nM T54771 CI17QE 89630302 EC50 = 3049 nM T54771 C7U8EF 89630310 EC50 = 874 nM T54771 CE90NZ 89630336 EC50 = 3576 nM T54771 CKQ8Z5 89630356 EC50 = 8167 nM T54771 C68EIV 89634067 EC50 = 845 nM T54771 CCI4Y3 89634111 EC50 = 1859 nM T54771 CX82JF 90177831 IC50 = 15.4 nM T54771 CNZ3M2 90183119 IC50 = 48.2 nM T54771 C83KZC 90183140 IC50 = 2 nM T54771 C36FVE 90183231 IC50 = 2.9 nM T54771 C8L0ZD 90644321 IC50 > 90000 nM T54771 CJAW70 90644322 IC50 > 90000 nM T54771 CJR19O 90644323 IC50 > 90000 nM T54771 CZ09VO 90644324 IC50 > 90000 nM T54771 CJ9R8U 90644325 IC50 > 90000 nM T54771 C3OB6A 117642291 IC50 = 2.7 nM T54771 CO4ZI9 127033993 EC50 = 3813 nM T54771 CUF5W6 127034238 EC50 = 5758 nM T54771 C1QJ6A 127034239 EC50 = 4692 nM T54771 C7JQ6C 129237363 IC50 = 52600 nM T54771 C8EN9I 133081837 IC50 = 1.1 nM T54771 CG36NB 133081841 IC50 = 1.6 nM T54771 CE26QS 133081845 IC50 = 8.4 nM T54771 CMI40H 133081848 IC50 = 6.8 nM T54771 CQC09F 133081850 IC50 = 14.8 nM T54771 C3ZMR2 133081853 IC50 = 1.7 nM T54771 C95PDI 134469373 IC50 = 3000 nM T54771 C5DF3L 134469421 IC50 = 2200 nM T54771 CIB5Y9 134469475 IC50 = 6400 nM T54771 CTN7F9 134469574 IC50 = 4800 nM T54771 C81HPB 134469603 IC50 = 25900 nM T54771 CDH70Y 134469622 IC50 = 4700 nM T54771 C2HV3Z 134469646 IC50 = 3600 nM T54771 C9U6KQ 134498364 IC50 = 5 nM T54771 C23TUN 134498374 IC50 = 32 nM T54771 C9C4XT 134498382 IC50 = 58 nM T54771 CX7R1U 134498384 IC50 = 39 nM T54771 CW4PQ9 134498385 IC50 = 33 nM T54771 CA2CX7 134498386 IC50 = 45 nM T54771 CX2V6Z 134498389 IC50 = 4 nM T54771 C1N6ZV 134498411 IC50 = 32 nM T54771 CA6TY7 134498420 IC50 = 5 nM T54771 CS3B7E 134498427 IC50 = 92 nM T54771 CC89KP 134498441 IC50 = 3 nM T54771 CD1F3O 134498886 IC50 = 3 nM T54771 C68VKL 134498938 IC50 = 206 nM T54771 C5M9BA 134498971 IC50 = 18 nM T54771 C8SWJ0 134499046 IC50 = 48 nM T54771 C41NYJ 134499051 IC50 = 84 nM T54771 C2DS4E 134512337 IC50 = 53 nM T54771 C6PO4L 135360405 IC50 = 5000 nM T54771 CLK6D0 135360457 IC50 = 2000 nM T54771 CZB1S9 135360458 IC50 = 22300 nM T54771 CK8DB1 135360478 IC50 = 500 nM T54771 CZ6Q2E 135360662 IC50 = 400 nM T54771 C3BN6R 135360764 IC50 = 400 nM T54771 CD90SA 135360772 IC50 = 1000 nM T54771 CG91HF 137498460 IC50 = 1421 nM T54771 CI9N6P 137498470 IC50 = 43 nM T54771 CP7R6L 137498479 IC50 = 376.1 nM T54771 C13MYJ 137498490 IC50 = 86 nM T54771 CXSR57 137498494 IC50 = 162.7 nM T54771 CTK58A 137498501 IC50 = 40.4 nM T54771 C76OXI 137498531 IC50 = 14 nM T54771 C5AZW2 137498544 IC50 = 186.6 nM T54771 CC0R7B 137498561 IC50 = 100.9 nM T54771 C89URP 137498572 IC50 = 96.4 nM T54771 CBR3V7 137631975 IC50 = 11600 nM T54771 CB1H9S 137635111 IC50 = 10600 nM T54771 CUFC09 137638493 IC50 = 235 nM T54771 C8RQG4 137639691 IC50 = 1082 nM T54771 CO03BT 137639897 IC50 = 14600 nM T54771 CNFX93 137640414 IC50 = 15100 nM T54771 C4R5MT 137647890 IC50 = 9700 nM T54771 C87NEV 137652303 IC50 = 453 nM T54771 CJMB48 137655785 IC50 = 13800 nM T54771 C2ZA4G 137661404 IC50 = 15600 nM T54771 CY92AB 137661679 IC50 = 31000 nM T54771 CBNS65 140930597 IC50 = 500 nM T54771 CQ9MJ6 145979226 IC50 = 414 nM T54771 C2XS9K 145980077 IC50 = 51 nM T54771 CTC03M 145980886 IC50 = 32 nM T54771 C2MC3U 145981567 IC50 = 35 nM T54771 CP96KA 145983611 IC50 > 10000 nM T54771 CQ5JG2 145983720 IC50 > 10000 nM T54771 C27EKA 145984945 IC50 > 10000 nM T54771 C7QIM1 145986927 IC50 = 22 nM T54771 C0NIQ8 145989102 IC50 = 47 nM T54771 CZM3G5 145989671 IC50 = 35 nM T54771 CUP18S 145992935 IC50 = 156 nM T54771 C7QD1G 155511498 IC50 = 55 nM T54771 C62GZS 155512672 IC50 = 55 nM T54771 C0Y6AF 155513930 IC50 = 34 nM T54771 CXS5V9 155519466 IC50 = 1166 nM T54771 CRLS07 155520018 IC50 = 21 nM T54771 CPKH72 155521866 IC50 = 22 nM T54771 C0L3BR 155527667 IC50 = 12531 nM T54771 CW9E6G 155527919 IC50 = 23 nM T54771 CGQF25 155529209 IC50 = 176 nM T54771 C6QYU8 155534804 IC50 = 111 nM T54771 C4Z3YH 155555849 IC50 = 36 nM T54771 C8FX9U 155556004 EC50 = 330 nM T54771 CDB31T 155559931 IC50 = 34 nM T54771 C2L5VQ 155568482 IC50 = 74 nM T54771 D00HFT 46229075 IC50 = 4000 nM T54771 D01DIQ 46229072 IC50 = 39000 nM T54771 D03AJS 10177526 IC50 = 2300 nM T54771 D05AZW 46229071 IC50 = 44000 nM T54771 D06WAL 6072 IC50 = 60.7 nM T54771 D0H6DA 11949247 IC50 = 2.1 nM T54771 D0HD2G 4788 IC50 = 12400 nM T54771 D0I2FC 15837283 IC50 = 50000 nM T54771 D0K6SV 44560286 IC50 = 0.17 nM T54771 D0L8OJ 45269680 IC50 = 5000 nM T54771 D0M8EH 45488072 IC50 = 1300 nM T54771 D0Q2YH 44560285 IC50 = 2 nM T54771 D0VE0Q 72936 IC50 = 18700 nM T54771 D0X1TN 9824918 IC50 = 22000 nM T85115 CX15AZ 11950138 IC50 = 461 nM T85115 CHR2Z9 11950301 IC50 > 10000 nM T85115 CKV42F 11950302 IC50 = 336 nM T85115 C1ZQB3 11950304 IC50 = 2500 nM T85115 C8JP2Q 11950479 IC50 = 2180 nM T85115 CRH17V 11950660 IC50 = 33 nM T85115 C8EW9Q 11950852 IC50 = 3690 nM T85115 C1VJW4 11950853 IC50 > 10000 nM T85115 C32BTM 11951031 IC50 = 19 nM T85115 CNX67F 11951384 Ki = 22 nM T85115 C8ID2M 11952097 IC50 = 51 nM T85115 CW79XH 11952273 IC50 = 318 nM T85115 C17YPD 25138121 Ki = 440 nM T85115 C0ZH5A 25138122 Ki = 4719 nM T85115 CI67EQ 45267221 IC50 = 2860 nM T85115 C0ZH5G 45267225 IC50 = 6510 nM T85115 C2NLF3 45268077 IC50 = 21 nM T85115 CMY49V 45269806 IC50 = 22 nM T85115 C5OQ9E 45269815 IC50 = 27 nM T85115 C2QYH5 45269816 IC50 = 1870 nM T85115 CC8A0H 45270634 IC50 = 1210 nM T85115 C0DT2H 45270642 IC50 = 3260 nM T85115 C6L9OJ 45272352 IC50 = 1160 nM T85115 C43HUP 45272355 IC50 = 4780 nM T85115 CEB1G6 45272370 IC50 = 47 nM T85115 COTE10 45273221 IC50 = 2590 nM T85115 CI73XU 45273238 IC50 > 10000 nM T85115 CRY4B6 45273239 IC50 = 515 nM T85115 CVB85E 91799673 IC50 = 290 nM T85115 C9S8MX 118111803 IC50 > 9000 nM T85115 C1F0RQ 118111817 IC50 = 320 nM T85115 CZHL82 118111824 IC50 = 910 nM T85115 C32FIN 118111843 IC50 = 7410 nM T85115 CWV5Z6 118120155 IC50 = 330 nM T69506 D06NXY 5991 IC50 = 3000 nM T69506 D09GOS 2812 Ki = 100 nM T69506 D0VN4K 1345 IC50 = 390 nM T69506 CKP1A6 71264 IC50 = 4078 nM T69506 C0HN5G 449196 IC50 = 1200 nM T69506 CJ79PF 798455 IC50 > 70000 nM T69506 C2B9IV 969470 IC50 = 687 nM T69506 CCU7V8 1008292 IC50 = 5010 nM T69506 C4KJF3 1069332 IC50 = 38755 nM T69506 C74ECK 1069342 IC50 = 235 nM T69506 CU4L6I 1129891 IC50 = 620 nM T69506 CXH30E 1129894 IC50 = 6400 nM T69506 C4VAP8 1129896 IC50 > 70000 nM T69506 C1ZYP7 1129899 IC50 = 320 nM T69506 C2IW9M 1129900 IC50 = 2430 nM T69506 C0JMB3 1212773 IC50 = 288 nM T69506 CH2TN3 1380478 IC50 = 3631 nM T69506 C0CAD6 1380480 IC50 = 1792 nM T69506 CG71XT 1645708 IC50 = 24490 nM T69506 CCUL28 9633071 EC50 = 580 nM T69506 CTE1N2 24748569 EC50 > 10000 nM T69506 CR5SI0 44476535 EC50 > 10000 nM T69506 CJ3FM4 46925833 EC50 = 2070 nM T69506 CUD91T 49862248 EC50 > 10000 nM T69506 CG1L3D 110168287 IC50 = 210 nM T69506 C17LEA 110168295 IC50 = 249 nM T69506 CKB6P7 110168297 IC50 = 680 nM T69506 CPX74Y 127027105 IC50 = 4080 nM T69506 CG5O2F 127027106 IC50 = 1410 nM T69506 C4OT8R 127027107 IC50 = 39810 nM T69506 C3UI4V 127028360 IC50 = 21.2 nM T69506 CTUD46 127028363 IC50 = 152.9 nM T69506 CAN20J 127028364 IC50 = 216.2 nM T69506 CVZK27 127028365 IC50 = 116 nM T69506 CFAV80 127028366 IC50 = 11.7 nM T69506 CQ2RG9 127028689 IC50 = 81.5 nM T69506 C5A8NT 127028690 IC50 = 37.6 nM T69506 C91ZAK 127028691 IC50 = 19.5 nM T69506 CI46GB 127028692 IC50 = 24.1 nM T69506 CYU2V6 127028696 IC50 = 31.9 nM T69506 CU90JV 127028697 IC50 = 22.1 nM T69506 C10WFX 127028698 IC50 = 20.1 nM T69506 C70GRE 127038883 IC50 = 13.9 nM T69506 CHUF28 127038906 IC50 = 3180 nM T69506 C0ME6N 127040363 IC50 = 37 nM T69506 CUKA16 127040364 IC50 = 2060 nM T69506 CGFV68 127040386 IC50 = 70.8 nM T69506 CRAP86 127040387 IC50 = 2320 nM T69506 CC23IJ 127040700 IC50 = 1030 nM T69506 C3CH6S 127040701 IC50 = 14420 nM T69506 C75EKQ 127040702 IC50 = 4930 nM T69506 C9CQO2 127040703 IC50 = 12970 nM T69506 C6UK2N 127041180 IC50 = 6890 nM T69506 CYX61D 127041941 IC50 = 13990 nM T69506 CVU05R 127042259 IC50 = 19090 nM T69506 CF6PO1 127042260 IC50 = 18790 nM T69506 CRF03T 127042261 IC50 = 116.4 nM T69506 C3C9IW 127042607 IC50 = 20.9 nM T69506 CDHR34 127042608 IC50 = 11350 nM T69506 CHTI58 127042609 IC50 = 60.1 nM T69506 CO8LH1 127042610 IC50 = 35.3 nM T69506 CNF97G 127042639 IC50 = 3050 nM T69506 C0U6OQ 127042934 IC50 = 1580 nM T69506 CI3X9L 127049803 EC50 = 690 nM T69506 C2O5LX 127049804 EC50 = 4040 nM T69506 C3BOI2 142505355 EC50 = 480 nM T69506 C2ICN5 142505357 EC50 = 740 nM T69506 CD41PR 142505358 EC50 = 10000 nM T69506 C2DHC6 142505361 EC50 = 670 nM T69506 CMLP67 142505363 EC50 = 1600 nM T69506 C9ZK0J 142505364 EC50 = 650 nM T69506 CCF42T 142505365 EC50 = 2400 nM T69506 C6KV3Z 142505366 EC50 = 490 nM T69506 CO7EZ3 142505367 EC50 = 940 nM T69506 C3QKF0 142505369 EC50 = 670 nM T69506 CCX3N7 142505373 EC50 = 920 nM T69506 C01EXB 142505375 EC50 = 10000 nM T69506 CK2R1S 142505382 EC50 = 460 nM T69506 CG4ZE8 142505390 EC50 = 1700 nM T69506 CELM50 142505396 EC50 = 980 nM T69506 CLB7T6 142505400 EC50 = 2600 nM T69506 C42FHG 142505403 EC50 = 150 nM T69506 CI5KU7 142505405 EC50 = 9200 nM T69506 C7WMR4 142505416 EC50 = 2100 nM T69506 CW4XY3 142505419 EC50 = 380 nM T69506 C4D0JN 142505420 EC50 = 400 nM T69506 C5B8OK 142505421 EC50 = 370 nM T69506 CF2QD5 142505424 EC50 = 2100 nM T69506 CAE56P 142505426 EC50 = 2200 nM T69506 CWU2V6 142505427 EC50 = 1500 nM T69506 CA7O9B 142505428 EC50 = 63000 nM T69506 CXTL63 142505432 EC50 = 660 nM T69506 CVC97Z 142505433 EC50 = 2700 nM T69506 CHB93R 142505434 EC50 = 840 nM T69506 CX8UP1 142505435 EC50 = 1900 nM T69506 C2MX6O 142505438 EC50 = 3400 nM T69506 CH1OC4 142505439 EC50 = 3200 nM T69506 C49CMN 142505442 EC50 = 440 nM T69506 CRV6K9 142505445 EC50 = 470 nM T69506 CH61LA 142505446 EC50 = 1500 nM T69506 CE8K7S 142505448 EC50 = 990 nM T69506 C09VYQ 142505449 EC50 = 2800 nM T69506 CS3E2Y 142505451 EC50 = 1500 nM T69506 CYOT59 142505454 EC50 = 190 nM T69506 C71NAW 142505463 EC50 = 410 nM T69506 CL3T1N 142505465 EC50 = 1100 nM T69506 CH1WB6 142505467 EC50 = 54000 nM T69506 CKD38I 142505471 EC50 = 8700 nM T69506 CUZ5E2 142505477 EC50 = 240 nM T69506 CZQR32 142505480 EC50 = 490 nM T69506 CHEO79 142505481 EC50 = 1100 nM T69506 C0TBH5 142505484 EC50 = 930 nM T69506 C73LTV 142505488 EC50 = 1100 nM T69506 C4GX9V 142505496 EC50 = 1300 nM T69506 C2AG0C 142505500 EC50 = 880 nM T69506 CJP7K4 142505503 EC50 = 560 nM T69506 CE6C3B 142505504 EC50 = 1100 nM T69506 C1JBX3 155269230 EC50 = 4400 nM T69506 CLF8Z4 155524131 EC50 > 100000 nM T69506 C29IZQ 155533563 EC50 = 590 nM T69506 CO7CM0 155535509 EC50 = 7900 nM T69506 D01BXE 9600409 EC50 = 20 nM T04388 D0I2FI 2993 IC50 = 1300 nM T04388 CV4Q5S 704452 IC50 = 4 nM T04388 C9MD5I 704533 IC50 > 30000 nM T04388 CQ6L4F 704624 IC50 > 30000 nM T04388 CL95TM 746607 IC50 > 30000 nM T04388 CDK30S 772885 IC50 = 25 nM T04388 C23RUP 873000 IC50 > 30000 nM T04388 CM27DN 954216 IC50 > 30000 nM T04388 CSR03N 11587013 EC50 = 400 nM T04388 CR40EH 23373327 IC50 > 30000 nM T04388 C67LUP 24857841 IC50 = 3000 nM T04388 C2UY6M 24946933 EC50 = 20 nM T04388 C6CZ1L 25110719 IC50 = 350 nM T04388 C8PXJ3 44393382 IC50 = 60 nM T04388 CV87IP 44578863 IC50 > 30000 nM T04388 CAM4V5 44579554 IC50 > 30000 nM T04388 CQ31VC 44579555 IC50 > 30000 nM T04388 CX75RU 44579608 IC50 > 30000 nM T04388 CJ2AK1 44589880 IC50 = 1100 nM T04388 C5KZ6N 44589881 IC50 = 19100 nM T04388 CL6F5D 44589882 IC50 = 14600 nM T04388 CNF98X 44589883 IC50 > 30000 nM T04388 C8XES0 44589884 IC50 = 15900 nM T04388 C6SX2P 44589885 IC50 = 10000 nM T04388 CM34HP 44589886 IC50 = 5200 nM T04388 C75WMJ 44589936 IC50 = 10700 nM T04388 C6H1GS 44589937 IC50 = 14600 nM T04388 C37JNX 44589938 IC50 = 11000 nM T04388 C6AE5U 44589939 IC50 = 7900 nM T04388 CH81DN 44589940 IC50 > 30000 nM T04388 CBO24P 44589941 IC50 > 30000 nM T04388 C9B6CX 44589988 IC50 > 30000 nM T04388 CZD26X 44589989 IC50 = 15400 nM T04388 C6NI7G 44589990 IC50 > 30000 nM T04388 CQT1V6 44589991 IC50 > 30000 nM T04388 CJC6U2 44589992 IC50 > 30000 nM T04388 CKY3S6 44589993 IC50 > 30000 nM T04388 C2E4HB 44590042 IC50 = 1000 nM T04388 C1O7IF 44590043 IC50 = 7500 nM T04388 CWC04O 57390845 Ki = 1268 nM T04388 C4C3RA 57396284 Ki = 837 nM T04388 C0U3HP 57401348 Ki = 46 nM T04388 CL5MG9 57403100 Ki = 575 nM T04388 CN0P9L 57403256 Ki = 214 nM T04388 C6STI3 72198633 IC50 = 31 nM T04388 D0H4BF 25102784 EC50 = 1810 nM T00612 D00SQN 12136798 IC50 = 110 nM T00612 D01QIN 60823 IC50 = 22547 nM T00612 D06WTZ 53232 IC50 = 25933 nM T00612 D09DHY 6167 IC50 > 20 ug.mL-1 T00612 D0E3SH 6918837 Ki = 0.65 nM T00612 D0E7PQ 5311 Ki = 1.6 nM T00612 D0L7LC 5352062 Ki = 0.038 nM T00612 D0Y3KG 3121 IC50 = 62000 nM T00612 D00FHR 9865515 Ki = 32.4 nM T00612 D01WKZ 53340426 IC50 = 318 nM T00612 D05KED 53340666 IC50 = 48 nM T00612 D06TKI 49857317 IC50 = 4 nM T00612 D07FPY 6918877 Ki = 36 nM T00612 D09XIZ 11538455 Ki = 0.06 nM T00612 D0B3FV 6445533 Ki = 1.4 nM T00612 D0B7CH 4775 IC50 = 65000 nM T00612 D0E6UZ 54575456 IC50 = 1.6 nM T00612 D0GE5B 56654642 IC50 = 1280 nM T00612 D0GH3Q 9804992 Ki = 3 nM T00612 D0L2UQ 49855250 Ki = 16 nM T00612 D0M8FD 4261 Ki = 65 nM T00612 D0V0SL 11749858 Ki = 19 nM T00612 D0XT6W 6918638 Ki = 0.85 nM T00612 D0Z4RC 24756910 IC50 = 12.6 nM T00612 D0J8OC 5186 Ki = 2.2 nM T00612 D00HXJ 118884610 Ki = 774 nM T00612 D0CH8Q 56965342 IC50 = 30 nM T00612 D0L1NO 72722126 IC50 > 50000 nM T00612 D0N2DK 72710871 IC50 = 8 nM T00612 D0QX3G 71532921 IC50 = 4400 nM T00612 D0YN2T 86302836 IC50 > 50000 nM T00612 D0ZG5X 71811260 IC50 = 3610 nM T00612 D0N3SH 4996 Ki = 36000 nM T00612 D0W9NH 2746 IC50 = 147 nM T00612 CBIR94 10313 IC50 = 7910 nM T00612 C1N2KZ 88129 IC50 = 680000 nM T00612 CW70DI 211808 IC50 > 100000 nM T00612 CF60JA 220184 IC50 > 33330 nM T00612 CE45SU 247630 IC50 > 1000 nM T00612 CH1JD3 419176 IC50 = 9000 nM T00612 C0Y4WC 614947 Ki = 0.42 nM T00612 CU3HS2 1108280 IC50 > 100000 nM T00612 C96GFC 1798422 IC50 = 100500 nM T00612 C94IXC 2173124 IC50 = 8750 nM T00612 C58NGX 2175719 IC50 = 6450 nM T00612 CJCY71 2295078 IC50 = 3020 nM T00612 CG41FO 2423676 IC50 = 5350 nM T00612 CEO31B 2423687 IC50 = 5860 nM T00612 CK8I3T 3432579 IC50 > 33330 nM T00612 CZA83Y 4118131 IC50 = 2720 nM T00612 CV9JS5 4288771 IC50 > 33000 nM T00612 CN4M6D 5281220 IC50 = 38900 nM T00612 CSIJ53 5793932 IC50 = 5100 nM T00612 C2NA1H 5842785 IC50 > 5000 nM T00612 C18ENP 6918846 Ki = 39 nM T00612 C1RD7E 6918878 Ki = 1.5 nM T00612 CE9LP2 9543539 IC50 = 1590 nM T00612 CJ07ZA 9800555 IC50 = 160 nM T00612 CC0EU7 9828788 IC50 = 3.9 nM T00612 CH2LR4 9835152 IC50 = 381 nM T00612 CLYJ85 9848223 IC50 = 270 nM T00612 CSW4Y1 9891541 IC50 = 200 nM T00612 C81EYJ 9923508 IC50 = 3 nM T00612 CQG4V8 9924543 IC50 = 0.8 nM T00612 COLN58 9965621 IC50 = 607 nM T00612 CQDG65 10110195 IC50 = 200 nM T00612 CWA9R2 10135838 IC50 = 441 nM T00612 CL4C9H 10154438 Ki = 0.1 nM T00612 C7RC1E 10309899 IC50 = 9 nM T00612 C9OU5F 10464879 Ki = 0.13 nM T00612 CDY91S 10584105 Ki = 0.26 nM T00612 CSMT47 10728039 Ki = 0.81 nM T00612 CK8UV7 11019840 Ki = 0.06 nM T00612 C5P3EI 11167060 IC50 = 80 nM T00612 C8G5WP 11210533 IC50 = 9100 nM T00612 CYJ60V 11244651 IC50 = 16400 nM T00612 CI7W3O 11267278 IC50 = 6460 nM T00612 CM6ZW2 11279156 IC50 = 4640 nM T00612 CY34EQ 11393847 IC50 = 200 nM T00612 CB3N5M 11514394 IC50 = 321 nM T00612 CRZ7H2 11556677 IC50 = 18 nM T00612 C2F9NT 11558827 IC50 = 647 nM T00612 C9UN7F 11637884 IC50 = 14500 nM T00612 C24SBP 11657529 IC50 = 160 nM T00612 CQ32FV 11664499 IC50 = 4 nM T00612 CG9OC4 11682502 IC50 = 17.9 nM T00612 CYB26W 11688197 IC50 > 1000 nM T00612 CJ2UA0 11690271 IC50 = 3360 nM T00612 CC3GQ0 11700059 IC50 = 59 nM T00612 CU0M1E 11947684 IC50 = 3.9 nM T00612 C0QCW4 11988293 IC50 = 2300 nM T00612 C9G1BN 11993595 IC50 = 3900 nM T00612 CH5JS7 11993694 IC50 = 440 nM T00612 CJ94OC 12542182 Ki > 2500 nM T00612 C06UTF 13507024 IC50 = 16 nM T00612 C4XJ8M 13889849 Ki = 470 nM T00612 C1KR4L 14113324 IC50 > 50000 nM T00612 C15MQN 14113325 IC50 > 50000 nM T00612 C2D1KP 15983982 Ki = 21 nM T00612 C7DK5L 15984110 IC50 = 500 nM T00612 CHB82E 15986417 IC50 = 2640 nM T00612 C52EVH 15986418 IC50 = 590 nM T00612 C0GED2 15986506 IC50 = 220 nM T00612 CEL7P9 15986507 IC50 = 460 nM T00612 CS1QO9 15986509 IC50 = 1160 nM T00612 C5T1WF 16006672 IC50 = 313 nM T00612 CQGC05 16036765 IC50 = 170 nM T00612 CM3T2E 16049824 IC50 = 29 nM T00612 C30UFT 16066811 IC50 = 272 nM T00612 CFK8J5 16068056 Ki = 26 nM T00612 CMQP70 16068495 Ki = 33 nM T00612 CT84XO 16068594 Ki = 18 nM T00612 CF3ZG5 16068595 Ki = 18 nM T00612 CL60CA 16068912 Ki = 14 nM T00612 C9ZQB3 16095102 Ki > 5000 nM T00612 C80XYC 16095113 Ki > 5000 nM T00612 C6BGM2 16659535 IC50 = 460 nM T00612 CQI9N3 16659537 IC50 = 330 nM T00612 C5YFV9 16661453 IC50 = 1480 nM T00612 C8S5OX 16661455 IC50 = 560 nM T00612 CH67WF 16661458 IC50 = 460 nM T00612 CZ72YC 16661613 IC50 = 260 nM T00612 C8DZ1T 16661615 IC50 = 1480 nM T00612 CQV40I 16661617 IC50 = 1440 nM T00612 C5CIB4 16663079 IC50 = 640 nM T00612 CUG50I 16733294 IC50 = 156 nM T00612 CWO7V0 16733295 IC50 = 2580 nM T00612 C4W0PG 16733410 IC50 = 167 nM T00612 C0MO3Z 16733411 IC50 = 113 nM T00612 C3QL4X 16733412 IC50 > 30000 nM T00612 CV54SY 16733414 IC50 = 1250 nM T00612 C1VCX2 16733415 IC50 = 492 nM T00612 CXN07K 16733416 IC50 > 30000 nM T00612 CP9AR8 16733417 IC50 = 205 nM T00612 CUE62T 16733590 IC50 > 30000 nM T00612 CB4IN2 16773791 IC50 = 2200 nM T00612 CQHD27 20459443 IC50 = 1050 nM T00612 CE2W3M 21630365 IC50 = 4800 nM T00612 CS5R0U 22836624 Ki = 12500 nM T00612 CD16PI 23521584 IC50 = 330 nM T00612 CB8A5Q 23648260 IC50 = 6 nM T00612 C1JZ6D 23648261 IC50 = 100 nM T00612 CQJS61 23648262 IC50 = 60 nM T00612 C35ILE 23648263 IC50 = 70 nM T00612 C82BVC 23648264 IC50 > 10000 nM T00612 CT6NY2 23648265 IC50 > 10000 nM T00612 CZV0Q2 23648266 IC50 = 60 nM T00612 C36NKL 23648268 IC50 = 200 nM T00612 C5YBX0 23760408 IC50 = 5000 nM T00612 CM73VT 23818230 IC50 = 2.1 nM T00612 CVAB64 23846833 IC50 = 3600 nM T00612 C8RC9P 24744325 IC50 = 45 nM T00612 CVB7J3 24746434 IC50 = 44 nM T00612 C28AWJ 24746436 IC50 = 71 nM T00612 C17GDO 24779722 IC50 >= 50 nM T00612 CA7O1E 24779723 IC50 >= 50 nM T00612 CIO7Q6 24853792 IC50 = 880 nM T00612 CBN0J5 24853793 IC50 = 110 nM T00612 CLT5J2 24881257 IC50 = 679 nM T00612 C5GCM1 24881328 IC50 = 294 nM T00612 C8QVB1 24881329 IC50 = 143 nM T00612 CU0AM3 24881330 IC50 = 43 nM T00612 CQM51L 24881331 IC50 = 63.9 nM T00612 C4KH8F 24881332 IC50 = 57.4 nM T00612 C1KA3V 24881333 IC50 = 216 nM T00612 C47APB 24881402 IC50 = 112 nM T00612 CSN8W1 24881403 IC50 = 167 nM T00612 C1UQ3K 24881404 IC50 = 47.5 nM T00612 C51TMH 24881405 IC50 = 77.4 nM T00612 C9EZI7 24881406 IC50 = 64.4 nM T00612 C6P3HS 24881407 IC50 = 124 nM T00612 CZ3TU1 24881464 IC50 = 146 nM T00612 CDI49N 24881465 IC50 = 124 nM T00612 CQGP87 24881466 IC50 = 116 nM T00612 CS1MH8 24888322 IC50 = 29000 nM T00612 CC0R9O 24938735 IC50 = 9.5 nM T00612 CF03HD 24948905 IC50 = 1740 nM T00612 CHP8O6 24948906 IC50 = 56.7 nM T00612 C1KRT8 24948907 IC50 = 1940 nM T00612 CKY2P8 24948908 IC50 = 147 nM T00612 C25CFI 24948909 IC50 = 1050 nM T00612 CWQ04Z 24948910 IC50 = 131 nM T00612 CM9I3X 24951310 IC50 = 133 nM T00612 CX1YF8 24951311 IC50 = 1690 nM T00612 CV10XU 24951312 IC50 = 238 nM T00612 CD6KV0 24951313 IC50 = 2980 nM T00612 CQY9Z0 24951314 IC50 = 93 nM T00612 CV8EF6 25032862 IC50 = 13 nM T00612 C35POS 25065102 IC50 >= 50 nM T00612 C62CND 25065309 IC50 >= 50 nM T00612 CNQ9O6 25065932 IC50 >= 50 nM T00612 CYC81K 25066135 IC50 >= 50 nM T00612 CZO9K3 25066136 IC50 >= 50 nM T00612 CH1Q5J 25066137 IC50 >= 50 nM T00612 CXD04I 25066140 IC50 = 500 nM T00612 CDF80L 25066350 IC50 = 500 nM T00612 CCKR19 25066353 IC50 >= 50 nM T00612 CX69SY 25066355 IC50 = 1930 nM T00612 CF8VP4 25066356 IC50 = 1570 nM T00612 CS9XH7 25066547 IC50 = 1540 nM T00612 C46AGN 25066548 IC50 = 207 nM T00612 CJF2M7 25066549 IC50 = 793 nM T00612 C7ZN2W 25118059 IC50 = 2.1 nM T00612 C4I1CJ 25155417 IC50 = 72 nM T00612 C72PBH 25155955 IC50 = 740 nM T00612 CB4E2J 25155956 IC50 = 71 nM T00612 CP4C5Y 25157071 IC50 = 470 nM T00612 CO14XG 25195084 IC50 = 140 nM T00612 C6BDX3 25207860 IC50 = 189000 nM T00612 CCD5M7 25227504 IC50 = 158 nM T00612 CK0D5S 25227505 IC50 = 382 nM T00612 CN97JP 25227508 IC50 = 268 nM T00612 CW8R1B 25227513 IC50 = 425 nM T00612 CE0NV4 25257993 IC50 = 4.39 nM T00612 C43BHY 25269097 IC50 = 54 nM T00612 CJ1RQ7 42598706 IC50 = 5160 nM T00612 C2LES7 42599455 IC50 = 3.1 nM T00612 C2KO0F 42599456 IC50 = 2.5 nM T00612 C1UAO7 42601485 IC50 = 14 nM T00612 CU23PG 42611301 IC50 = 5 nM T00612 CW1G2R 42611390 IC50 = 40 nM T00612 C62QFJ 42611486 IC50 = 70 nM T00612 CQ37HN 42612743 IC50 = 3.38 nM T00612 CX1UT9 42612744 IC50 = 825.2 nM T00612 CXK4C1 42618298 IC50 = 5 nM T00612 CQB20M 42630929 IC50 = 1700 nM T00612 CN93YB 42630930 IC50 > 5000 nM T00612 CH7RW1 42630932 IC50 = 450 nM T00612 CC8B0M 42630933 IC50 > 5000 nM T00612 CDT65Y 42631047 IC50 > 5000 nM T00612 CH69CQ 42631048 IC50 = 1200 nM T00612 C2NF6U 42632370 IC50 = 320 nM T00612 C2EA1T 42632371 IC50 = 310 nM T00612 C69LCN 42632491 IC50 = 1200 nM T00612 C9B8VR 42632614 IC50 > 5000 nM T00612 CB79DG 42637299 IC50 = 3600 nM T00612 CP36KB 42637300 IC50 > 100000 nM T00612 CI8J6H 42637372 IC50 = 530 nM T00612 C5RYO0 42637373 IC50 > 100000 nM T00612 CJ0CG5 42638004 IC50 = 99000 nM T00612 C8X0TG 42638005 IC50 = 830 nM T00612 CO57GS 44138033 IC50 = 15800 nM T00612 CQ2VD5 44219634 IC50 = 164 nM T00612 CY0QB9 44253226 IC50 = 270 nM T00612 CZ8R1N 44253780 IC50 = 192 nM T00612 C7G5CO 44359547 IC50 = 890 nM T00612 CIT7A9 44359548 IC50 = 41000 nM T00612 CUM0Q6 44359555 IC50 = 5900 nM T00612 CP92JV 44359673 IC50 > 100000 nM T00612 CQ7J2G 44359674 IC50 = 7800 nM T00612 CGK71T 44359675 IC50 = 11000 nM T00612 C2V4DN 44359681 IC50 = 1400 nM T00612 CX31TB 44359788 IC50 = 19000 nM T00612 CQ5Y8G 44359800 IC50 > 100000 nM T00612 CL82CH 44359814 IC50 > 100000 nM T00612 C5YRC9 44431499 IC50 = 110000 nM T00612 CK2P0J 44443716 IC50 = 500 nM T00612 CQ1WD9 44443718 IC50 = 500 nM T00612 CNC51G 44447194 IC50 = 105 nM T00612 C5VP4D 44454144 IC50 = 360 nM T00612 CJ0L4C 44456965 IC50 = 170 nM T00612 C74LTB 44506448 IC50 = 33 nM T00612 CPDE25 44507029 IC50 = 6300 nM T00612 C2UZ1P 44507247 IC50 = 560 nM T00612 CBL69N 44507542 IC50 = 20000 nM T00612 C7F8YJ 44543715 Ki = 125 nM T00612 CIO34V 44564642 Ki = 39 nM T00612 CG9OD1 44571302 IC50 = 520 nM T00612 C0ZX1A 44571330 IC50 = 5540 nM T00612 CY83MO 44571331 IC50 = 1810 nM T00612 CP6D1G 44571332 IC50 = 3470 nM T00612 CMA3R6 44574139 IC50 = 430 nM T00612 C5KLR7 44574177 IC50 > 30000 nM T00612 CFS49I 44574178 IC50 > 30000 nM T00612 CJ32DK 44574179 IC50 > 30000 nM T00612 CQOS28 44574180 IC50 = 469 nM T00612 CN96ZV 44574181 IC50 = 3750 nM T00612 CWJA85 44574206 IC50 > 30000 nM T00612 C46XHW 44574207 IC50 > 30000 nM T00612 C3RY9V 44574208 IC50 > 30000 nM T00612 CT7F0N 44589856 IC50 = 110 nM T00612 CA6Q9Y 44592060 IC50 = 13200 nM T00612 C5H8RA 44598536 IC50 = 290 nM T00612 CC2QV9 44623002 IC50 > 50000 nM T00612 CVJ51M 44623152 IC50 > 50000 nM T00612 C6TJ2G 44623153 IC50 > 50000 nM T00612 C8I7GL 44818075 IC50 > 1000 nM T00612 C42SJP 45141750 IC50 = 239 nM T00612 CLE9U5 45141751 IC50 = 589 nM T00612 CSM1O6 45271073 IC50 = 1100 nM T00612 C2M4GV 46179732 IC50 = 27.5 nM T00612 CS75CD 46179779 IC50 = 25.1 nM T00612 C39YKM 46179780 IC50 = 48.2 nM T00612 C0CKE5 46180624 IC50 > 30000 nM T00612 C7GYH0 46180758 IC50 = 60 nM T00612 C27IKH 46180759 IC50 = 24.6 nM T00612 CSC1Y9 46180760 IC50 = 28.5 nM T00612 C70FSJ 46180763 IC50 = 27.8 nM T00612 C0W8DB 46187719 IC50 = 1630 nM T00612 CV7D4Z 46187885 IC50 = 920 nM T00612 C53ZSX 46187886 IC50 = 8150 nM T00612 CEV52J 46187887 IC50 = 1580 nM T00612 CSC70G 46187888 IC50 = 8560 nM T00612 C7SC8A 46187889 IC50 = 2790 nM T00612 CQLG06 46187890 IC50 = 4530 nM T00612 CVGN05 46187891 IC50 = 7320 nM T00612 CF29IN 46188075 IC50 = 1050 nM T00612 COWJ59 46190552 IC50 > 10000 nM T00612 C8YO4W 46190553 IC50 > 10000 nM T00612 CEX48K 46190554 IC50 > 10000 nM T00612 C6J9DI 46190555 IC50 = 7690 nM T00612 C53RNX 46190556 IC50 > 10000 nM T00612 CPS37G 46190557 IC50 = 8520 nM T00612 C2MOT0 46190609 IC50 = 9230 nM T00612 CJ8OT2 46190610 IC50 > 10000 nM T00612 CX93ZQ 46190753 IC50 = 1170 nM T00612 C85WSJ 46190754 IC50 > 10000 nM T00612 C9VEX6 46190755 IC50 = 5190 nM T00612 C6O5AD 46190756 IC50 = 230 nM T00612 C7F8AM 46190820 IC50 = 7930 nM T00612 C8JY0S 46190821 IC50 = 1250 nM T00612 CUCK61 46190822 IC50 = 1560 nM T00612 CXQ51Y 46190823 IC50 = 2780 nM T00612 CR0G9O 46190824 IC50 = 390 nM T00612 CDP80X 46190825 IC50 = 510 nM T00612 C3ETP2 46190826 IC50 = 6260 nM T00612 CD57RJ 46197798 IC50 = 31 nM T00612 CR04HA 46197799 IC50 = 48 nM T00612 CQ83FI 46203315 IC50 = 730 nM T00612 CK8YL5 46203316 IC50 = 680 nM T00612 C1YB9P 46203618 IC50 = 3850 nM T00612 C4I5DH 46203619 IC50 > 10000 nM T00612 C43KVC 46203620 IC50 = 6290 nM T00612 CY7ER9 46203621 IC50 > 10000 nM T00612 CW13ZY 46203622 IC50 > 10000 nM T00612 CND31M 46203623 IC50 = 5190 nM T00612 C1RX2K 46203949 IC50 = 3160 nM T00612 CZJ86R 46203950 IC50 = 2870 nM T00612 CNA07J 46203951 IC50 = 2570 nM T00612 CQ69AM 46205433 IC50 = 165 nM T00612 CQTI31 46881225 IC50 > 30000 nM T00612 CVDH51 46887335 IC50 = 10000 nM T00612 CPS5F8 46887435 IC50 = 21000 nM T00612 CJ26EB 46887436 IC50 = 10000 nM T00612 CZP2B8 46887476 IC50 = 3800 nM T00612 C25DSY 46887918 IC50 = 179 nM T00612 C93CLK 46887919 IC50 = 11400 nM T00612 CPSI47 46890583 Ki = 12 nM T00612 C90NYX 46896338 IC50 = 250 nM T00612 CAT34L 46906643 IC50 = 90400 nM T00612 C4V7PG 46907052 IC50 = 10400 nM T00612 CMQ3R0 46907054 IC50 = 16500 nM T00612 C2PC1Z 46907160 IC50 = 96300 nM T00612 C1HV6U 46907409 IC50 = 20 nM T00612 CXH64A 46918825 IC50 = 25118.86 nM T00612 C6GY9I 46934544 IC50 = 18900 nM T00612 C3OD2Y 46934546 IC50 = 36200 nM T00612 CH61CW 47187185 IC50 > 1000 nM T00612 CL7PS1 49831258 IC50 > 50000 nM T00612 CI5L2P 49846123 IC50 = 563.7 nM T00612 C4DL0M 49847150 IC50 = 128 nM T00612 CC7Y9U 49850262 IC50 = 360 nM T00612 C50PXU 49855444 IC50 > 50000 nM T00612 C6POK9 49856931 IC50 = 14 nM T00612 C52ABG 50942502 IC50 = 290 nM T00612 CPQ0F7 50991199 IC50 = 29 nM T00612 COA5W3 51051073 IC50 = 82 nM T00612 C8U2AI 51180076 IC50 > 1000 nM T00612 CV76KB 51357270 IC50 = 72 nM T00612 CE43FC 53249967 IC50 > 30000 nM T00612 C7MO2J 53325871 IC50 = 26.5 nM T00612 CG84JS 53325976 IC50 = 800 nM T00612 CVM4Q3 53357987 IC50 = 3900 nM T00612 C78GKN 53361474 IC50 = 1000 nM T00612 CNB63X 53361475 IC50 = 780 nM T00612 CQ43VH 53363518 Ki = 8.6 nM T00612 C6Y2EV 53374826 IC50 = 6360 nM T00612 C9U7GF 53464577 IC50 = 4 nM T00612 C4EYP7 53464578 IC50 = 361.8 nM T00612 C0WNH9 53464579 IC50 = 199.4 nM T00612 C4MQ3U 53464638 IC50 = 2.3 nM T00612 CJ53ZV 53464639 IC50 = 381.1 nM T00612 CN9RH2 53464770 IC50 = 189.3 nM T00612 C5A7MU 54613496 IC50 = 34.1 nM T00612 CJ1G6K 56591671 IC50 = 670 nM T00612 CIO96M 56659403 IC50 > 100000 nM T00612 C7R9TZ 56663191 IC50 = 0.9 nM T00612 CL18NI 56666337 IC50 > 100000 nM T00612 C9LC5Y 56673234 IC50 > 100000 nM T00612 CWH5N4 56673261 IC50 > 100000 nM T00612 C2ML5S 56837168 IC50 = 20.4 nM T00612 CCW89V 56932477 IC50 = 1.11 nM T00612 CZ25SN 56935695 IC50 > 30000 nM T00612 CP4EL2 57328394 IC50 = 28000 nM T00612 CW02FD 57393108 IC50 = 740 nM T00612 CX0I2Z 57396604 IC50 = 880 nM T00612 CB8N4P 57400091 IC50 = 800 nM T00612 C5CRJ1 57412107 IC50 = 320 nM T00612 COG4Q8 57412108 IC50 = 190 nM T00612 C4LI0D 57521296 IC50 = 31000 nM T00612 CXFJ46 57550498 IC50 = 2700 nM T00612 CWT6O0 57723146 IC50 = 140 nM T00612 CA5Q6O 58147189 IC50 > 50000 nM T00612 C4DYC0 58147224 IC50 > 50000 nM T00612 CMP04X 58147302 IC50 > 50000 nM T00612 CLD40J 58465708 IC50 = 39000 nM T00612 C1MB4Q 59323957 IC50 > 30000 nM T00612 CK6LX0 59454220 IC50 = 220 nM T00612 C2SDN1 59454252 IC50 = 270 nM T00612 CO6A2S 59585196 IC50 = 710000 nM T00612 CLN20W 60143424 IC50 = 39.6 nM T00612 CEF0C3 60143425 IC50 = 43.6 nM T00612 CRNZ07 60145504 IC50 = 38.2 nM T00612 C31TUG 60145641 IC50 = 44.1 nM T00612 CG6M7H 60145642 IC50 = 3.9 nM T00612 C8XKG0 60145643 IC50 = 45.2 nM T00612 CC72HW 60145644 IC50 = 46.6 nM T00612 CBHR24 60145645 IC50 = 40.7 nM T00612 CS85AJ 60145783 IC50 = 48.1 nM T00612 C8SZ7X 60145784 IC50 = 5.2 nM T00612 CIP62A 60145785 IC50 = 45.5 nM T00612 CZPN39 60145786 IC50 = 48.5 nM T00612 CGX45C 60145787 IC50 = 40.3 nM T00612 CPZ5Q3 60148646 IC50 > 50000 nM T00612 C8ZL3J 60148690 IC50 > 50000 nM T00612 CK5N4E 60148693 IC50 = 43000 nM T00612 CB7X2E 60151224 IC50 = 45 nM T00612 CY05OU 60151225 IC50 = 328 nM T00612 CWO8H0 60152596 IC50 = 2710 nM T00612 CXW14A 60164619 IC50 = 12589.25 nM T00612 C5F0OQ 62706003 IC50 = 210 nM T00612 CQAM69 62706004 IC50 = 3200 nM T00612 C6CK5L 62706005 IC50 = 2400 nM T00612 C08BWT 62706006 IC50 = 10000 nM T00612 COTB68 62706167 IC50 = 830 nM T00612 CM0LI9 62706168 IC50 = 750 nM T00612 C5I8OL 62706169 IC50 = 77000 nM T00612 CW48QK 62706170 IC50 = 1000 nM T00612 CIQ52T 62706171 IC50 = 350 nM T00612 C8V2NC 62706321 IC50 = 1000 nM T00612 CBN3L0 69950064 Ki > 19000 nM T00612 C6RFQ8 70676597 IC50 > 20000 nM T00612 CD0YC8 70681968 IC50 = 4870 nM T00612 CM62BN 70682297 IC50 = 1580 nM T00612 CH2OA7 70684090 IC50 = 4990 nM T00612 C60XID 70684091 IC50 = 1150 nM T00612 C8L6YP 70686231 IC50 = 570 nM T00612 CGJK81 70686232 IC50 = 1150 nM T00612 CWF4E8 70688346 IC50 = 5020 nM T00612 CTE30H 70690378 IC50 = 6520 nM T00612 C7VF1B 70692849 Ki = 33 nM T00612 C28UMB 70693708 IC50 = 32 nM T00612 C1JO8E 70694590 IC50 = 2670 nM T00612 CWJ39I 70694591 IC50 = 2360 nM T00612 CE67KO 70695508 IC50 = 3300 nM T00612 C3DW5T 70696631 IC50 = 2170 nM T00612 CD5O7B 70696632 IC50 = 550 nM T00612 CQY1I6 70789579 Ki > 19000 nM T00612 CQ2E6U 71142135 IC50 = 3680 nM T00612 C8NZA0 71449818 IC50 = 72000 nM T00612 C63AHI 71449819 IC50 = 79000 nM T00612 C3J9QZ 71453454 IC50 = 1200 nM T00612 C57ATO 71455172 IC50 = 2000 nM T00612 C6B2HJ 71456958 IC50 = 300 nM T00612 CM9A3I 71458827 IC50 = 370 nM T00612 C72DJO 71465631 IC50 = 62 nM T00612 C0CX7P 71476624 Ki = 0.22 nM T00612 C6QPH1 71476625 Ki = 0.04 nM T00612 C3JLD4 71476626 Ki = 0.12 nM T00612 C3OH6T 71476627 Ki = 0.51 nM T00612 C0LWJ6 71520631 IC50 = 1392 nM T00612 CO28HI 71520716 IC50 = 944 nM T00612 CVA5Q7 71520717 IC50 = 881 nM T00612 C89SWX 71527724 IC50 > 30000 nM T00612 C6S5JQ 71527847 IC50 = 321.6 nM T00612 C6KBD4 71534512 IC50 = 1900 nM T00612 CT51EW 71534810 IC50 = 60 nM T00612 C7QN3O 71534812 IC50 = 15 nM T00612 C8M3HU 71537640 IC50 = 2230 nM T00612 C2QML7 71537641 IC50 = 37 nM T00612 CU0ZE6 71537928 IC50 = 78 nM T00612 CH9FS7 71537929 IC50 = 601 nM T00612 CTW95A 71537931 IC50 = 48 nM T00612 C3C0RO 71538475 IC50 = 70 nM T00612 CIA28E 71538746 IC50 = 67 nM T00612 CFCV26 71538748 IC50 = 2540 nM T00612 CY2T1Q 71538749 IC50 = 1770 nM T00612 C4A6VJ 71538750 IC50 = 68 nM T00612 CG72NC 71538751 IC50 = 168 nM T00612 C7RUE6 71540743 IC50 = 32100 nM T00612 C9LA4F 71540744 IC50 = 3880 nM T00612 C0EK5J 71540745 IC50 = 30800 nM T00612 C80HZX 71540746 IC50 = 224 nM T00612 C5UZQ0 71540747 IC50 = 25100 nM T00612 C4G5US 71540862 IC50 = 3270 nM T00612 CDW81Y 71574856 IC50 = 16790 nM T00612 CX01BJ 71574948 IC50 = 341 nM T00612 CO8YU7 71574949 IC50 = 1610 nM T00612 CBZ5S9 71583103 IC50 = 26000 nM T00612 C3PSJ9 71583105 IC50 = 29000 nM T00612 C21GHR 71624738 IC50 = 1200 nM T00612 CU65GH 71655059 IC50 = 657.7 nM T00612 CPS58L 71655136 IC50 = 468.3 nM T00612 CFW7Q9 71655137 IC50 = 414.2 nM T00612 C9S0UB 71655138 IC50 = 467.2 nM T00612 CU27EV 71655139 IC50 = 600.1 nM T00612 CO8R1Z 71655216 IC50 = 463.3 nM T00612 C0W6EK 71655283 IC50 = 881.8 nM T00612 C7HG0K 71655802 IC50 = 1790 nM T00612 CPJ4V7 71680913 IC50 = 9000 nM T00612 C9X8KM 71680914 IC50 = 20000 nM T00612 C4W2MA 71680915 IC50 = 11000 nM T00612 C3KO9V 71680916 IC50 = 30000 nM T00612 CN4X5O 71680917 IC50 > 33000 nM T00612 CWAM13 71680918 IC50 > 33000 nM T00612 CI9G3B 71681069 IC50 = 4800 nM T00612 CFUC24 71722010 IC50 = 111.2 nM T00612 CEG67K 71723449 IC50 = 1120 nM T00612 CTSK68 71811225 IC50 = 6450 nM T00612 C1K6OW 71811226 IC50 = 4000 nM T00612 CU3N9R 71811227 IC50 = 1610 nM T00612 CS2L4B 71811228 IC50 = 2210 nM T00612 CL4DT9 71811229 IC50 = 1220 nM T00612 CK6DB4 71811230 IC50 > 12000 nM T00612 CHR8V0 71811259 IC50 = 4810 nM T00612 CVL54T 71811261 IC50 > 10000 nM T00612 CZR93K 71811262 IC50 = 6880 nM T00612 CM8BE4 71811290 IC50 = 4780 nM T00612 C0MV3O 71811291 IC50 > 10000 nM T00612 C7UYD4 71811292 IC50 = 7480 nM T00612 C7XL3N 71811293 IC50 > 10000 nM T00612 C4HBC5 71811294 IC50 > 10000 nM T00612 CTA26S 71811295 IC50 = 5680 nM T00612 C9GHU8 71818097 IC50 = 111 nM T00612 CAW2Q1 71818098 IC50 = 81 nM T00612 CE89AK 71818242 IC50 = 580 nM T00612 C8M3IX 71818243 IC50 = 920 nM T00612 CKP5J7 71818244 IC50 = 440 nM T00612 CT7L6G 72163687 Ki = 0.25 nM T00612 CKE9D3 72163688 Ki = 0.23 nM T00612 CI9H6L 72164895 IC50 = 231 nM T00612 CS5UL7 72195322 IC50 = 397 nM T00612 CAC5Q7 72375561 IC50 = 1300 nM T00612 C3WQV2 72375562 IC50 = 20 nM T00612 CC1W6J 72375670 IC50 = 2100 nM T00612 CY8R0O 72696205 IC50 = 10390 nM T00612 C56QXM 72696206 IC50 = 53520 nM T00612 C0CM8Q 72696335 IC50 = 140 nM T00612 C73XOU 72734382 IC50 = 1150 nM T00612 CJR6C9 72734542 IC50 = 770 nM T00612 CV09DJ 72734543 IC50 = 3.5 nM T00612 CS6LW0 72946640 IC50 = 89 nM T00612 CXM37Z 72946641 IC50 = 142 nM T00612 CQA16N 72946833 IC50 = 143 nM T00612 CNR7Z2 72946834 IC50 = 689 nM T00612 C12JYS 72946835 IC50 = 238 nM T00612 C5Y9XH 72946836 IC50 = 110 nM T00612 CVZR94 72946837 IC50 = 5040 nM T00612 C8-AUG 72946838 IC50 = 956 nM T00612 CHQ39Y 72947043 IC50 = 143 nM T00612 CCST90 72947044 IC50 = 27 nM T00612 C7J3RH 72947045 IC50 = 93 nM T00612 CK10LZ 73292342 IC50 > 12000 nM T00612 CX3W1T 73333311 IC50 = 16000 nM T00612 CDG47J 73346009 IC50 > 20000 nM T00612 C6H7IJ 73346010 IC50 > 20000 nM T00612 CD0WU2 73346011 IC50 > 20000 nM T00612 COBJ19 73347538 IC50 = 1430 nM T00612 C92HFB 73349064 IC50 > 20000 nM T00612 C68LBO 73349131 IC50 = 21 nM T00612 CAS8E2 73352138 IC50 > 20000 nM T00612 C0C2QO 73353595 IC50 > 20000 nM T00612 C59WMZ 73353596 IC50 = 16700 nM T00612 C1UDF8 73353597 IC50 = 248 nM T00612 CUD02X 73355098 IC50 = 134 nM T00612 CXK86S 73355189 IC50 = 193 nM T00612 CD6L5K 73707349 IC50 = 1 nM T00612 C26KZD 73707535 IC50 = 6.9 nM T00612 CM1H3U 73707536 IC50 = 18.8 nM T00612 CH97TE 73707543 IC50 = 14.2 nM T00612 C2PWQ3 73707544 IC50 = 21 nM T00612 CEM5B6 73707545 IC50 = 6.3 nM T00612 CPQ43R 73707550 IC50 = 10.8 nM T00612 CJ1DA8 73774764 IC50 = 498.5 nM T00612 CQ3K6G 73776326 IC50 = 535.5 nM T00612 CC4L0G 73776327 IC50 = 432.1 nM T00612 CZB6G7 73776472 IC50 = 498.1 nM T00612 CSRE84 73776614 IC50 = 457 nM T00612 C01FVX 73776616 IC50 = 413.6 nM T00612 C3UC9H 73891099 IC50 = 10000 nM T00612 CM6H9C 76324878 IC50 > 50000 nM T00612 CL4JQ3 76331862 IC50 = 4390 nM T00612 C08CPW 76335428 IC50 = 180 nM T00612 C7JQU3 76335755 IC50 = 5840 nM T00612 CKI74A 76853213 IC50 > 20000 nM T00612 CCR7L2 76853289 IC50 > 100000 nM T00612 CJ6Z0X 78324068 IC50 > 20000 nM T00612 C3U0KE 81689842 IC50 > 50000 nM T00612 CG5ZD9 86291495 IC50 = 8.2 nM T00612 C61VCD 86294741 IC50 = 400000 nM T00612 CBWV30 86294747 IC50 = 95000 nM T00612 C06YBD 86302594 IC50 = 9490 nM T00612 C3EM7H 86581004 IC50 = 20 nM T00612 C7UK3Y 86581005 IC50 = 93 nM T00612 CY64UM 86581152 IC50 = 18 nM T00612 CY5V7C 86581153 IC50 = 10 nM T00612 C1HE8I 86581432 IC50 = 100 nM T00612 CZM07I 86581434 IC50 = 22 nM T00612 C8ZQG9 86581435 IC50 = 25 nM T00612 C6M9PL 86765212 IC50 = 1160 nM T00612 CS5I4Y 87261507 IC50 = 160 nM T00612 CQ2LF5 88920533 IC50 > 10000 nM T00612 CP1NA9 89183138 IC50 = 156 nM T00612 CQS6C0 89183185 IC50 = 219 nM T00612 CWY3H6 90024758 IC50 > 1000 nM T00612 CSBC45 90024759 IC50 > 1000 nM T00612 CB73DR 90025023 IC50 > 1000 nM T00612 C5P3DT 90025027 IC50 > 1000 nM T00612 C9GB2A 90025255 IC50 > 1000 nM T00612 C5W0UY 90025331 IC50 > 1000 nM T00612 C7NHW6 90025915 IC50 > 1000 nM T00612 CRC9B5 90026100 IC50 > 1000 nM T00612 CR53ON 90026278 IC50 > 1000 nM T00612 CX2U6G 90063981 IC50 > 1000 nM T00612 CZB49Y 90063982 IC50 > 1000 nM T00612 C8RG2T 90064049 IC50 > 1000 nM T00612 C2YQM7 90064053 IC50 > 1000 nM T00612 C62GSL 90654859 IC50 = 791.2 nM T00612 CJH1S6 90654947 IC50 > 10000 nM T00612 C94IWR 90654948 IC50 > 10000 nM T00612 CSR56C 90655296 IC50 = 5610 nM T00612 CSDO81 90664458 Ki = 27 nM T00612 CAQL21 91667420 IC50 = 69.8 nM T00612 C5M9AK 91667421 IC50 = 20.77 nM T00612 CJO6T1 91810840 IC50 = 2200 nM T00612 CYJ12Q 91884636 IC50 = 78 nM T00612 C34WIG 92045024 IC50 > 100000 nM T00612 C9OC0F 101882265 IC50 = 109000 nM T00612 CDV40P 101882454 IC50 = 160 nM T00612 C2I8XR 101882814 Ki = 1400 nM T00612 CVE07R 101882857 IC50 = 2230 nM T00612 C63EWT 101882858 IC50 = 3290 nM T00612 C8KZB4 101883993 Ki = 900 nM T00612 C7Q6ID 101884982 IC50 = 33 nM T00612 CR46PQ 101884983 IC50 = 34 nM T00612 CRZ83C 101884989 IC50 = 171 nM T00612 CT7Z8F 102514716 IC50 > 10000 nM T00612 CS2UL0 117829456 IC50 = 170 nM T00612 C7L4OT 117829461 IC50 = 100 nM T00612 C50VUN 117829462 IC50 = 90 nM T00612 CH27PR 118613747 IC50 = 21 nM T00612 C0OX4M 118613748 IC50 = 1.1 nM T00612 CNF09H 118613750 IC50 = 150 nM T00612 C3ETI2 118613751 IC50 = 3.1 nM T00612 C9KZQ0 118613755 IC50 = 1.4 nM T00612 C30OPU 118613756 IC50 = 6.3 nM T00612 C46TFD 118613757 IC50 = 1.4 nM T00612 C1J5AG 118613783 IC50 = 1.7 nM T00612 C9T0ML 118613821 IC50 = 1.1 nM T00612 CSU52M 118656852 IC50 > 30000 nM T00612 CB6AJ9 118656853 IC50 > 30000 nM T00612 C45UYG 118709095 IC50 = 33000 nM T00612 C7QHE4 118712502 IC50 = 0.5 nM T00612 C8KSD6 118712503 IC50 = 0.9 nM T00612 C1JFZ7 118714371 IC50 = 2747 nM T00612 CXF0U3 118714375 IC50 = 558 nM T00612 C2M5OR 118714376 IC50 = 204 nM T00612 CY4GN9 118714377 IC50 = 226 nM T00612 CM5QT7 118719376 Ki = 1700 nM T00612 CPB7C3 118719377 Ki = 600 nM T00612 C09OGH 118719378 Ki = 400 nM T00612 CR5VC1 118719379 Ki = 800 nM T00612 C32LCM 118719380 Ki = 300 nM T00612 C8U6YR 118719381 Ki = 300 nM T00612 C9Y0HV 118719382 Ki = 300 nM T00612 CY0J4D 118719383 Ki = 300 nM T00612 CCYU59 118719817 IC50 = 12 nM T00612 CSC47W 118720522 IC50 = 864.5 nM T00612 CUI51W 118720529 IC50 = 64.8 nM T00612 CCGH73 118720703 IC50 = 16400 nM T00612 CMV2W9 118721625 IC50 = 28 nM T00612 CF5TO3 118721859 IC50 = 103 nM T00612 CK97TZ 118721860 IC50 = 13 nM T00612 CYV30O 118721861 IC50 = 14 nM T00612 C5WYI1 118721862 IC50 = 5 nM T00612 CSMW25 118721863 IC50 = 6640 nM T00612 C5B1KM 118721864 IC50 = 454 nM T00612 CG8LZ0 118721865 IC50 = 19400 nM T00612 CPCN23 118721866 IC50 = 14000 nM T00612 CM0A9U 118721867 IC50 = 10700 nM T00612 C8IAG9 118734664 IC50 = 10420 nM T00612 CJ6KL7 118734665 IC50 = 380 nM T00612 C2VQ5P 118734666 IC50 = 4910 nM T00612 CYF71E 118734667 IC50 = 190 nM T00612 CQC7H0 118734668 IC50 = 6730 nM T00612 CP27CN 118734669 IC50 = 270 nM T00612 CBIY72 118734670 IC50 > 20 ug.mL-1 T00612 C9C7UX 118734705 IC50 = 5410 nM T00612 C16OUT 118735146 IC50 = 530 nM T00612 CZRV81 118735147 IC50 = 560 nM T00612 CFE4D0 118735148 IC50 = 290 nM T00612 C97NHV 118735149 IC50 = 5930 nM T00612 CQ0FJ3 118735150 IC50 = 430 nM T00612 CD4J8E 118735151 IC50 = 150 nM T00612 C7UE8T 118735152 IC50 = 280 nM T00612 CS6WO5 118735153 IC50 = 4390 nM T00612 C4XZ3C 118735154 IC50 = 8370 nM T00612 CRL6V4 118735155 IC50 = 320 nM T00612 CI8G4X 118737400 IC50 = 1770 nM T00612 C2F8TQ 118737455 IC50 = 380.5 nM T00612 C1T6WZ 118738004 IC50 > 10000 nM T00612 CZ61KV 118753026 IC50 = 1500 nM T00612 CFI23Y 118753027 IC50 = 6000 nM T00612 C75LTK 118753189 IC50 = 27000 nM T00612 C8DVP1 118868599 Ki = 7244 nM T00612 C9G4LD 118868621 Ki = 234 nM T00612 CQT5I6 118868656 Ki = 6097 nM T00612 CE3PD1 118868670 Ki > 10000 nM T00612 C5L8QM 118884518 IC50 = 3340 nM T00612 CV0E3L 118884590 Ki = 484 nM T00612 CME8R7 118884591 Ki = 1356 nM T00612 C4XJ7F 118884592 Ki = 66.51 nM T00612 CP5TE9 118884676 Ki = 943 nM T00612 CVTL89 118884679 Ki = 370 nM T00612 CB84TO 121278998 IC50 > 50000 nM T00612 C9S5OK 121279020 IC50 > 50000 nM T00612 CL3M2F 121499152 IC50 = 168 nM T00612 C93JAV 122177622 IC50 = 255 nM T00612 C5HJ0C 122177623 IC50 > 10000 nM T00612 CSU97K 122177957 IC50 = 275 nM T00612 CR8WL1 122180003 IC50 > 10000 nM T00612 CW4K2U 122181880 IC50 = 349.5 nM T00612 CK63UH 122181881 IC50 = 655.4 nM T00612 C0H9WU 122181882 IC50 = 4.42 nM T00612 CR3TU6 122181883 IC50 = 471.8 nM T00612 C57VRL 122181884 IC50 = 1240 nM T00612 C9V6XI 122186483 IC50 = 270 nM T00612 CU74JP 122186484 IC50 = 180 nM T00612 C7M2EU 122186485 IC50 = 360 nM T00612 CCG1Z2 122186543 IC50 = 610 nM T00612 CI32QY 122186544 IC50 = 250 nM T00612 CBN3P1 122186553 IC50 = 192 nM T00612 CP83NA 122186554 IC50 = 94 nM T00612 CPN31F 122191258 IC50 > 5000 nM T00612 CL5WI0 122191259 IC50 > 5000 nM T00612 CRTN32 122191260 IC50 = 1050 nM T00612 C1ZRE6 122191261 IC50 > 5000 nM T00612 C97BGS 122191262 IC50 > 5000 nM T00612 C1GUZ3 122191263 IC50 > 5000 nM T00612 CJG60T 122191264 IC50 > 5000 nM T00612 C28JVO 122192004 IC50 = 36.6 nM T00612 CF2D8U 122192005 IC50 = 2740 nM T00612 CW1HK5 122195536 IC50 = 6.8 nM T00612 C5W8OZ 122376192 IC50 = 25.6 nM T00612 C3V5ND 122550211 IC50 = 386 nM T00612 C63EYP 122601008 IC50 > 3000 nM T00612 CCN03D 122601010 IC50 > 10000 nM T00612 CZC01M 122601076 IC50 > 3000 nM T00612 CZE35C 122648343 IC50 = 3.9 nM T00612 C54RNT 122648367 IC50 = 2.9 nM T00612 C1UVI7 122648600 IC50 = 11.46 nM T00612 CMX59K 122648648 IC50 = 2.62 nM T00612 CVZ64I 122648649 IC50 = 2.8 nM T00612 CJR97Y 123525532 IC50 > 1000 nM T00612 CVFI87 127025051 IC50 > 10000 nM T00612 CE4CI8 127025178 IC50 = 221 nM T00612 CM38EU 127025541 IC50 = 140 nM T00612 CY5T9P 127025646 IC50 > 3000 nM T00612 CKJ6L8 127025647 IC50 > 3000 nM T00612 C6D2IJ 127026516 IC50 = 165 nM T00612 C8BA3S 127027767 IC50 = 56 nM T00612 CG8NU7 127027995 IC50 = 72 nM T00612 CZ7C3D 127028030 IC50 = 3.3 nM T00612 CV07OM 127028943 IC50 = 68 nM T00612 CV9I8D 127030313 IC50 = 5200 nM T00612 CR0P1O 127031793 IC50 = 11800 nM T00612 C4GI0F 127037614 IC50 = 187 nM T00612 CSJ32V 127039213 IC50 = 154 nM T00612 CZ8A1F 127041696 IC50 = 29850 nM T00612 C5D2OJ 127044292 IC50 = 1450 nM T00612 C58KRZ 127044343 IC50 = 4730 nM T00612 C1TYS6 127044344 IC50 = 119 nM T00612 C3G0SM 127044498 IC50 = 1290 nM T00612 C5CP9M 127045259 IC50 = 6560 nM T00612 CB8HR2 129104138 IC50 > 50000 nM T00612 CCH65A 129104183 IC50 > 50000 nM T00612 CFH8Q4 129104227 IC50 > 50000 nM T00612 C6HM5P 129104349 IC50 > 50000 nM T00612 CZTF90 129104374 IC50 > 50000 nM T00612 CUJ2P5 129104402 IC50 > 50000 nM T00612 CY3I6X 129104426 IC50 > 50000 nM T00612 CGT6B0 130238385 Ki = 469 nM T00612 CMWV13 130238420 Ki = 310 nM T00612 C0GH4T 130238474 Ki = 70.8 nM T00612 C9ERM5 130238475 Ki = 768 nM T00612 C8IEV4 130258911 IC50 = 1870 nM T00612 CHVF85 132022730 IC50 > 100000 nM T00612 C6OXE3 132134663 IC50 = 49 nM T00612 CP8L7V 132137973 IC50 = 3103 nM T00612 C6X3HG 132145728 IC50 = 8610 nM T00612 C8O9DP 132157820 IC50 = 12500 nM T00612 C2N5JD 132279660 IC50 = 135 nM T00612 C4L6UZ 132547258 IC50 = 163 nM T00612 CGBR54 132547259 IC50 = 4050 nM T00612 CW4MP2 132547260 IC50 = 854 nM T00612 C1YO2Z 132547261 IC50 = 407 nM T00612 CU63DV 132569672 IC50 = 256 nM T00612 CIUZ08 132576538 IC50 = 439 nM T00612 CTE3A6 132576539 IC50 = 659 nM T00612 C87DPY 132576540 IC50 = 827 nM T00612 CG91UP 132576541 IC50 = 1788 nM T00612 CL2R5W 132576542 IC50 = 759 nM T00612 C5C2EQ 132576544 IC50 = 1294 nM T00612 CA5V0R 132576546 IC50 = 2915 nM T00612 C0Y2TP 132585192 IC50 = 66 nM T00612 C4KE3N 132938351 IC50 = 268 nM T00612 C4UAN3 134129876 IC50 = 294 nM T00612 C25EVA 134129883 IC50 = 302 nM T00612 CWRH43 134129994 IC50 = 232 nM T00612 CK2TM6 134130010 IC50 = 2060 nM T00612 CYW6H1 134130165 IC50 = 32 nM T00612 CQ7SN8 134131102 IC50 = 929 nM T00612 CQO23I 134131456 IC50 = 209 nM T00612 CHZ8A3 134131564 IC50 = 1360 nM T00612 CN9DL4 134132030 IC50 > 10000 nM T00612 CX93QK 134135812 IC50 > 100000 nM T00612 CN8L9J 134136160 IC50 = 580000 nM T00612 C53UTO 134137062 IC50 = 1100 nM T00612 CSX58U 134139437 IC50 = 3330 nM T00612 C08YTI 134140697 IC50 = 15 nM T00612 C75NRQ 134141877 IC50 > 100000 nM T00612 C62SVR 134142119 IC50 > 100000 nM T00612 CLI48U 134143743 IC50 = 14100 nM T00612 CUA26W 134143927 IC50 = 58000 nM T00612 CWRJ15 134147087 IC50 > 100000 nM T00612 C8K0XJ 134147090 IC50 = 3370 nM T00612 CQ61SB 134150479 IC50 = 86500 nM T00612 CDX75O 134152551 IC50 = 15000 nM T00612 C2JV5X 134153768 IC50 > 100000 nM T00612 C2E8MV 134154228 IC50 = 11.48 nM T00612 C38DIF 134156853 IC50 = 180000 nM T00612 C4FLQ5 134157355 IC50 > 100000 nM T00612 C1UP3S 134157845 IC50 = 2250 nM T00612 C0X1HQ 134224487 IC50 = 570 nM T00612 CZV43J 134283792 IC50 = 18000 nM T00612 C62WXO 134283796 IC50 = 51000 nM T00612 CO7K3N 134283799 IC50 = 4900 nM T00612 CBQ17L 134283800 IC50 = 36000 nM T00612 C1Y4TA 134283810 IC50 = 38000 nM T00612 CV2YF7 134283813 IC50 = 32000 nM T00612 C05FVT 134492522 IC50 > 10000 nM T00612 C52IBY 134823859 IC50 = 18000 nM T00612 CS1V6A 135367138 IC50 > 50000 nM T00612 CVO59N 135367789 IC50 > 50000 nM T00612 CDY18W 135407493 IC50 > 100000 nM T00612 CW2I4R 135412048 IC50 > 100000 nM T00612 C7U0AV 135412194 IC50 > 100000 nM T00612 CS54TL 135437514 IC50 = 67000 nM T00612 C36MUC 135441620 IC50 > 100000 nM T00612 CRB8M1 135444536 IC50 > 100000 nM T00612 CX5D6J 135446479 IC50 = 18900 nM T00612 C1TOK2 135449197 IC50 > 100000 nM T00612 CW25GL 135462117 IC50 > 100000 nM T00612 CCL28F 135473106 IC50 > 100000 nM T00612 CYA60G 135497781 IC50 > 100000 nM T00612 C01EZF 135567459 IC50 > 100000 nM T00612 CV3QP4 135886613 IC50 = 108 nM T00612 C8X5LO 135928012 Ki = 70 nM T00612 CI2YE8 135928628 IC50 > 100000 nM T00612 C50NIS 136025837 IC50 > 100000 nM T00612 C4OS0V 136025842 IC50 > 100000 nM T00612 CX7Z5B 136025843 IC50 > 100000 nM T00612 CB8EM9 136025984 IC50 > 100000 nM T00612 C49MUG 136025986 IC50 > 100000 nM T00612 C0OLS8 136030779 IC50 = 65000 nM T00612 CIA7R4 136030780 IC50 = 76000 nM T00612 C24LKN 136030781 IC50 > 100000 nM T00612 CH7Y3C 136086920 IC50 > 100000 nM T00612 C3VDL5 136086921 IC50 > 100000 nM T00612 C9GOB5 136086922 IC50 = 69300 nM T00612 CE3ZL7 136086923 IC50 > 100000 nM T00612 CJZ5F3 136086924 IC50 > 100000 nM T00612 CT19ND 136110961 IC50 = 110 nM T00612 CY9U0E 136173089 IC50 = 110 nM T00612 C19VDS 136237971 IC50 = 19200 nM T00612 CBS97C 136239447 IC50 = 85 nM T00612 CT2MI6 136239448 IC50 = 44 nM T00612 CE2F9G 136244081 IC50 = 56 nM T00612 C9CH7S 136244085 IC50 = 104 nM T00612 C5J2AX 136244086 IC50 = 82 nM T00612 C46CYT 136244087 IC50 = 425 nM T00612 CXY1L5 136244088 IC50 = 538 nM T00612 CILG36 136286746 IC50 = 117 nM T00612 C39WRP 136286747 IC50 > 20000 nM T00612 C7ZX5O 136286761 IC50 = 3860 nM T00612 C9SV6G 136645392 IC50 > 20000 nM T00612 CANQ56 136645396 IC50 > 20000 nM T00612 C9TGH1 136645397 IC50 > 20000 nM T00612 C1F7JV 136645401 IC50 > 20000 nM T00612 C32LNQ 136645404 IC50 = 14600 nM T00612 C4W0IE 136645405 IC50 > 20000 nM T00612 CMIU28 136645406 IC50 > 20000 nM T00612 C3K2WL 136645410 IC50 = 11400 nM T00612 CC1D0X 136645415 IC50 = 17500 nM T00612 C02RIK 136645417 IC50 > 20000 nM T00612 C8CT0Z 136645422 IC50 = 1110 nM T00612 CAWT82 136645431 IC50 = 1110 nM T00612 CBZ8Q1 136645433 IC50 > 20000 nM T00612 C21EJD 136645435 IC50 > 20000 nM T00612 C1KTV3 136645436 IC50 > 20000 nM T00612 CK1B9W 136645438 IC50 = 2550 nM T00612 C6QOP7 136645441 IC50 = 4800 nM T00612 CMZ71T 136645444 IC50 > 20000 nM T00612 CL47WS 136645445 IC50 = 799 nM T00612 C64BZR 136645447 IC50 > 20000 nM T00612 C7X1UL 136645449 IC50 = 1260 nM T00612 CI9ZO7 136645454 IC50 = 5190 nM T00612 CA3I8S 136645455 IC50 > 20000 nM T00612 CRN16W 136645457 IC50 = 1310 nM T00612 CGQ92L 136645458 IC50 = 6970 nM T00612 CO5DN2 136645462 IC50 = 4640 nM T00612 CRPN39 136645466 IC50 = 3720 nM T00612 CL5X3G 136645467 IC50 = 17500 nM T00612 C48HNY 136959539 IC50 = 1850 nM T00612 C1P8ZW 136959550 IC50 = 490 nM T00612 CKU95F 136966187 IC50 = 712 nM T00612 CFRG19 136985286 IC50 > 20000 nM T00612 CE7F4O 136985287 IC50 = 166 nM T00612 CFPT21 136985288 IC50 = 1940 nM T00612 CBH5Y0 136985291 IC50 = 2030 nM T00612 CDAK28 136985292 IC50 = 341 nM T00612 CQ9XW7 136985295 IC50 > 20000 nM T00612 C1M6NW 136985296 IC50 > 20000 nM T00612 CJOA28 136985302 IC50 = 4390 nM T00612 CE6QK0 137125258 IC50 = 160 nM T00612 CAW80Q 137125259 IC50 = 130 nM T00612 CP5NM4 137125260 IC50 = 280 nM T00612 C5CKZ8 137125261 IC50 = 180 nM T00612 C1ROQ9 137125262 IC50 = 290 nM T00612 CL29YN 137125263 IC50 = 180 nM T00612 C5OY8K 137125264 IC50 = 150 nM T00612 C0YGR6 137125265 IC50 = 240 nM T00612 CMYG96 137125266 IC50 = 340 nM T00612 CI78CK 137125267 IC50 = 230 nM T00612 CD62KP 137125268 IC50 = 400 nM T00612 CE8NM5 137125269 IC50 = 430 nM T00612 CANS59 137136982 IC50 > 20000 nM T00612 C5AE3Q 137283418 IC50 > 20000 nM T00612 C5QIX1 137289788 IC50 = 1860 nM T00612 C5X0YR 137289866 IC50 = 335 nM T00612 CU70ZB 137289868 IC50 > 20000 nM T00612 CV6AN7 137289892 IC50 > 20000 nM T00612 CB14CI 137289900 IC50 > 20000 nM T00612 CLY69S 137289946 IC50 > 20000 nM T00612 CC5HA4 137290225 IC50 > 20000 nM T00612 C4RBC7 137290234 IC50 > 20000 nM T00612 CKJ6Q4 137290238 IC50 > 20000 nM T00612 CR53GQ 137290273 IC50 = 490 nM T00612 C8DYG6 137290344 IC50 > 20000 nM T00612 C9G3JB 137292402 IC50 = 89 nM T00612 C6MXL3 137292504 IC50 = 6430 nM T00612 CAZ49O 137300702 IC50 = 1870 nM T00612 CGE0J6 137300703 IC50 = 13900 nM T00612 CDU43L 137300704 IC50 = 9830 nM T00612 CK0QG6 137300705 IC50 > 20000 nM T00612 C91IPL 137300706 IC50 > 20000 nM T00612 C5UYP8 137300707 IC50 > 20000 nM T00612 CHSG63 137300708 IC50 = 2250 nM T00612 CX57MR 137300709 IC50 = 14100 nM T00612 C54KGS 137300710 IC50 = 432 nM T00612 CQD07Z 137300711 IC50 > 20000 nM T00612 C3I1CB 137300712 IC50 > 20000 nM T00612 C9LP2B 137353123 IC50 = 1100 nM T00612 CNKJ27 137353141 IC50 = 1300 nM T00612 CAW4X1 137353146 IC50 = 3000 nM T00612 CAPH58 137353182 IC50 = 3200 nM T00612 CWM6Z2 137376574 Ki = 995 nM T00612 C3LUJ0 137487429 IC50 = 5300 nM T00612 CA5OY1 137628667 IC50 = 179 nM T00612 C67EFJ 137628684 IC50 = 0.61 nM T00612 CHL7E8 137631592 IC50 = 320 nM T00612 CJ7P1U 137631803 IC50 = 441 nM T00612 C1N8TU 137632249 Ki = 3195 nM T00612 C84MIY 137633138 IC50 = 337 nM T00612 CW8G1H 137633768 IC50 = 193.5 nM T00612 C82QCH 137633786 IC50 = 209.35 nM T00612 C73PDL 137634086 IC50 = 75 nM T00612 C1V8QE 137634156 IC50 = 6309.57 nM T00612 CZ1FK2 137635119 IC50 = 28.04 nM T00612 C6JVG9 137635398 IC50 = 5.8 nM T00612 CAWZ25 137635575 IC50 = 0.53 nM T00612 COF8J3 137635708 IC50 = 21.2 nM T00612 C2KS3O 137635975 IC50 = 3130 nM T00612 CK1S0F 137637029 IC50 = 3.9 nM T00612 CEI0W2 137637915 IC50 = 2500 nM T00612 CTUL07 137638741 IC50 = 0.9 nM T00612 CX8Q4R 137638837 Ki = 313 nM T00612 CDWG31 137638917 IC50 = 209 nM T00612 CUG0C9 137639328 IC50 > 10000 nM T00612 CJBF37 137639551 IC50 = 287.59 nM T00612 C3CD6L 137639796 IC50 = 2319.76 nM T00612 C06BYV 137640258 IC50 = 283.3 nM T00612 C19GDO 137640291 IC50 = 59.5 nM T00612 CS50ET 137641009 IC50 = 1340 nM T00612 C4OEC3 137641520 IC50 = 1300 nM T00612 C5JUR2 137641533 IC50 = 1040 nM T00612 C1PRH5 137642860 IC50 = 61 nM T00612 C37BJQ 137642900 IC50 = 194 nM T00612 CJOS87 137643760 IC50 = 223 nM T00612 C7DLO4 137644089 IC50 = 490 nM T00612 CCBN61 137645084 IC50 = 311 nM T00612 C8GNS5 137645287 IC50 = 3215.9 nM T00612 C8WPM4 137645400 IC50 = 1650 nM T00612 CX3E0H 137645675 IC50 = 121.3 nM T00612 C5REZ8 137645689 IC50 > 20000 nM T00612 CA0V2Q 137647353 IC50 = 146 nM T00612 CM65KH 137647813 IC50 = 0.18 nM T00612 CO7H5A 137648171 IC50 = 179 nM T00612 CN3I9X 137648982 IC50 = 111 nM T00612 C0PGD9 137649617 IC50 = 314 nM T00612 CGK2M9 137649620 IC50 = 90 nM T00612 CM15FY 137649624 IC50 > 10000 nM T00612 CEP9R0 137651700 IC50 = 970 nM T00612 CFLX25 137652000 IC50 = 2380 nM T00612 C8NHK9 137652359 IC50 > 5000 nM T00612 C5FHD3 137652442 IC50 = 20300 nM T00612 CMP7G0 137652638 IC50 = 121 nM T00612 CZI5S2 137653293 IC50 = 170 nM T00612 C3QX5N 137653295 IC50 = 332.1 nM T00612 CXZ5J3 137654094 IC50 = 84 nM T00612 CIW9C6 137654210 Ki = 5205 nM T00612 C3FEM8 137654512 IC50 = 1640 nM T00612 CCR5B3 137654793 IC50 = 47 nM T00612 C1SBN5 137654946 IC50 = 1408.14 nM T00612 C71ZNJ 137656226 IC50 > 10000 nM T00612 CVG9T3 137656290 IC50 = 26 nM T00612 C0NR1V 137656498 IC50 = 1460 nM T00612 CRP0T2 137656638 IC50 = 1270 nM T00612 C0EQI2 137656898 IC50 = 296 nM T00612 C76OGQ 137656942 IC50 = 24000 nM T00612 CY8A2I 137656945 IC50 = 88.77 nM T00612 C5BM7T 137657586 IC50 = 908 nM T00612 C97QUM 137657678 IC50 = 179 nM T00612 C21XDS 137657845 IC50 = 3500 nM T00612 CPJL30 137659007 IC50 = 217 nM T00612 C9D7NR 137659196 IC50 = 199.3 nM T00612 CFGW13 137659898 IC50 = 128 nM T00612 C6XWP9 137659968 IC50 = 385.51 nM T00612 CM0OE5 137660128 IC50 = 1120 nM T00612 CLWU57 137660171 IC50 = 191.3 nM T00612 CEJI95 137661885 IC50 = 69 nM T00612 CEF18M 137661927 IC50 > 5000 nM T00612 CAQ62X 137701235 Ki = 23 nM T00612 CXV84M 138377596 IC50 = 120 nM T00612 CIWG23 138393067 IC50 = 910 nM T00612 C7EM3I 138393071 IC50 = 568 nM T00612 C4NFS3 138393072 IC50 = 420.5 nM T00612 CA3C4O 138454792 IC50 = 3 nM T00612 CN2UH1 139303146 IC50 = 13.26 nM T00612 CN4M1E 139325532 IC50 = 2100 nM T00612 C9EBI4 139325820 IC50 = 8400 nM T00612 CP73QO 141504704 IC50 = 1260 nM T00612 C13JZX 141522811 IC50 = 47100 nM T00612 CHS9N0 141728829 IC50 = 730 nM T00612 C9H8PX 141728841 IC50 = 130 nM T00612 CBV2K5 141728842 IC50 = 190 nM T00612 C2HF9A 141728845 IC50 = 430 nM T00612 C4RGY1 141728867 IC50 = 1400 nM T00612 C7XI0V 141764754 IC50 = 3.6 nM T00612 CO6C7N 142489312 IC50 = 2800 nM T00612 C7B3JK 142489313 IC50 = 4800 nM T00612 CGT08I 142489314 IC50 = 1800 nM T00612 CF7K4G 142489316 IC50 = 2700 nM T00612 CM6LR2 142489318 IC50 = 2500 nM T00612 C42DBC 142489319 IC50 = 3000 nM T00612 CH5Y8E 142489322 IC50 = 1100 nM T00612 C5MN8W 142489323 IC50 = 2000 nM T00612 CFYC82 142489328 IC50 = 1200 nM T00612 C4DKW7 142489330 IC50 = 7800 nM T00612 CDS81U 142489335 IC50 = 630 nM T00612 CMY8W1 142489337 IC50 > 10000 nM T00612 CD5E9S 142489342 IC50 = 2000 nM T00612 C65LBI 142489344 IC50 = 3400 nM T00612 CX0E9B 142505968 IC50 = 14100 nM T00612 CBJC50 142505992 IC50 = 18190 nM T00612 C7N8LV 142506025 IC50 = 3247 nM T00612 CKBF56 142506033 IC50 = 1231 nM T00612 CGNQ74 142506189 IC50 = 7173 nM T00612 CP5HF8 142506225 IC50 = 25480 nM T00612 CF5CB6 144562551 IC50 > 1000 nM T00612 C0CRK4 144562558 IC50 > 1000 nM T00612 C5I0NG 144562573 IC50 > 1000 nM T00612 CDI1U5 144562574 IC50 > 1000 nM T00612 CDA28I 145949712 IC50 = 23 nM T00612 CXJ0Y4 145949850 IC50 = 20 nM T00612 C1EF9X 145950102 IC50 = 114 nM T00612 CRKM19 145950884 IC50 = 6.8 nM T00612 CV3QO5 145951170 IC50 = 999.6 nM T00612 CRSM78 145952088 IC50 = 32900 nM T00612 CFE4G6 145952135 IC50 = 263 nM T00612 CEC68O 145952295 IC50 = 4900 nM T00612 CKG98W 145953085 IC50 > 100000 nM T00612 CL0XT8 145954248 IC50 = 25 nM T00612 CM53ZB 145954785 IC50 = 10800 nM T00612 CNB9E6 145955015 IC50 = 4200 nM T00612 CGP9X1 145955496 IC50 = 232 nM T00612 CJ03TU 145957740 IC50 = 413 nM T00612 CBNG29 145957781 IC50 = 32 nM T00612 C3L8IE 145958641 IC50 = 1704 nM T00612 C8SI2G 145958925 IC50 > 10000 nM T00612 CO05IK 145959360 IC50 = 132 nM T00612 C9IV1C 145959866 IC50 = 33.1 nM T00612 CK1XI0 145960971 IC50 > 10000 nM T00612 C1X5EO 145962694 IC50 = 33 nM T00612 C29PAL 145963897 IC50 = 29000 nM T00612 CJ47DY 145964043 IC50 > 100000 nM T00612 C3PWD4 145964064 IC50 = 1950 nM T00612 CEX67F 145964240 IC50 = 47000 nM T00612 CEDK05 145964533 IC50 = 5500 nM T00612 CDO47P 145964554 IC50 = 40000 nM T00612 CDY56B 145964885 IC50 = 424 nM T00612 CB51JU 145965019 IC50 > 100000 nM T00612 CW6UM7 145965159 IC50 = 3100 nM T00612 C9XLE7 145966296 IC50 > 100000 nM T00612 CM6KY1 145966543 IC50 > 100000 nM T00612 CJAE67 145966594 IC50 = 7250 nM T00612 CTUF34 145966712 IC50 = 380 nM T00612 CTRI57 145966861 IC50 > 100000 nM T00612 CUD38A 145967089 IC50 = 2700 nM T00612 C19POY 145967140 IC50 = 5140 nM T00612 C93JKN 145967593 IC50 = 1974 nM T00612 CD82XB 145967610 IC50 = 135 nM T00612 C7OG1D 145967698 IC50 = 635 nM T00612 C5RPQ9 145967832 IC50 = 47 nM T00612 CI1ZD2 145967851 IC50 = 2883 nM T00612 CR59HK 145967905 IC50 = 883 nM T00612 C95SNQ 145967968 IC50 = 919 nM T00612 CES7W6 145968087 IC50 = 1503 nM T00612 CSO4I7 145968364 IC50 > 5000 nM T00612 CSJ81Y 145968726 IC50 = 1800 nM T00612 CG0S9U 145968824 IC50 = 763 nM T00612 CIA79M 145968985 IC50 = 114 nM T00612 C27YHM 145969456 IC50 = 40 nM T00612 CV53YN 145969651 IC50 = 391 nM T00612 C0K6XS 145969789 IC50 = 76 nM T00612 CZ80EP 145969996 IC50 = 1216 nM T00612 C79YOL 145970069 IC50 > 100000 nM T00612 CFL68X 145970091 IC50 > 100000 nM T00612 C7TSV2 145970161 IC50 = 1835 nM T00612 CG5OK8 145970171 IC50 = 42 nM T00612 C3FQ0V 145970292 IC50 = 11200 nM T00612 C8FXH4 145970309 IC50 = 99000 nM T00612 CBR60K 145970453 IC50 = 362 nM T00612 C0E2UO 145970598 IC50 = 17 nM T00612 CI43DY 145970786 IC50 = 1770 nM T00612 C7K1AJ 145971681 IC50 = 7472 nM T00612 CA0F3X 145972521 IC50 > 1000 nM T00612 CW0T7A 145973234 IC50 = 5740 nM T00612 CO51JK 145973368 IC50 = 98.8 nM T00612 C4HTO2 145973543 IC50 = 2140 nM T00612 CSR50O 145973656 IC50 = 70400 nM T00612 CFP2R3 145973876 IC50 > 100000 nM T00612 CVM0Z3 145974125 IC50 > 100000 nM T00612 CLCU89 145974270 IC50 = 5400 nM T00612 C8YEJ9 145974425 IC50 = 5110 nM T00612 CUJE21 145974558 IC50 > 10000 nM T00612 CY1G2F 145974565 IC50 = 491 nM T00612 C5YJO8 145974667 IC50 = 58000 nM T00612 CZL05M 145975187 IC50 > 100000 nM T00612 CE8I5V 145975869 IC50 = 4800 nM T00612 C6Y9QH 145975913 IC50 = 69000 nM T00612 CU65BZ 145976000 IC50 > 100000 nM T00612 C86GXV 145976671 IC50 = 13000 nM T00612 CMUA94 145976675 IC50 = 7270 nM T00612 CN6UO4 145977003 IC50 = 11600 nM T00612 CKAQ67 145977127 IC50 = 3030 nM T00612 C78XNS 145977336 IC50 > 100000 nM T00612 CLY4Z5 145977632 IC50 = 240 nM T00612 CP53JS 145977717 IC50 = 16.6 nM T00612 C3QYB8 145978561 IC50 > 100000 nM T00612 COR40V 145978805 IC50 = 2100 nM T00612 C7X4LZ 145978932 IC50 = 900 nM T00612 C0UG8S 145980171 IC50 = 390 nM T00612 CIM41N 145980574 IC50 = 410 nM T00612 CMB08D 145981960 IC50 = 147 nM T00612 CMY73B 145983639 IC50 = 6300 nM T00612 CWD0A9 145983712 Ki = 3.1 nM T00612 CB24HO 145985400 IC50 = 470 nM T00612 C56MWZ 145986208 Ki = 130 nM T00612 C1WH7V 145986586 IC50 > 5000 nM T00612 CS79CE 145986632 IC50 = 327 nM T00612 CRX8H1 145987492 IC50 = 41 nM T00612 CPAX89 145987732 IC50 = 40 nM T00612 CJ1M7T 145987832 IC50 = 6.6 nM T00612 CV3S8R 145988041 IC50 = 3230 nM T00612 C82CIN 145988785 IC50 > 30000 nM T00612 CJ8DO3 145989487 IC50 = 549 nM T00612 C68VKC 145993051 IC50 = 370 nM T00612 C1W6CF 145994016 IC50 = 12000 nM T00612 C0YXS8 147254231 IC50 = 4618 nM T00612 C48EXH 148289288 IC50 = 9.25 nM T00612 CN71OS 149405396 IC50 = 13620 nM T00612 CWG10H 151364732 IC50 = 97 nM T00612 C6I7OZ 152636346 IC50 = 85 nM T00612 C7LM4U 153534003 IC50 = 251 nM T00612 CP1V9H 153534004 IC50 = 105 nM T00612 C9FIY4 153534005 IC50 = 58 nM T00612 CVT63S 153534008 IC50 = 170 nM T00612 C7JFY3 154068925 IC50 > 1000 nM T00612 C0KW3O 155511274 IC50 = 174.6 nM T00612 C0LH8C 155511921 IC50 = 282 nM T00612 CB8RS9 155512087 IC50 > 25000 nM T00612 CV2MG0 155512401 IC50 = 81 nM T00612 CT4VS3 155512474 IC50 = 150 nM T00612 CQ5BL7 155512551 IC50 > 50000 nM T00612 C7VKU2 155513116 IC50 = 139 nM T00612 CHLO32 155513171 IC50 = 1300 nM T00612 C5WUJ6 155513192 IC50 = 112 nM T00612 CE4H7I 155513471 IC50 > 50000 nM T00612 CCDH73 155514314 IC50 = 5400 nM T00612 C6BV9W 155514532 IC50 = 1240 nM T00612 CW3VT9 155514603 IC50 > 50000 nM T00612 CZ84WI 155515284 IC50 > 50000 nM T00612 CWEZ05 155515488 IC50 = 2.46 nM T00612 CUKG21 155515602 IC50 > 50000 nM T00612 CYJ53T 155515864 IC50 = 8100 nM T00612 C1K2XN 155516139 IC50 = 4942 nM T00612 CRS8L2 155516458 IC50 > 1000 nM T00612 CA1J3N 155517086 IC50 = 249 nM T00612 CL72ME 155517175 IC50 = 49.5 nM T00612 C7G0XM 155517418 IC50 = 4100 nM T00612 CY54TU 155518062 IC50 > 30000 nM T00612 CEH2N5 155518106 IC50 = 277 nM T00612 C58ZNC 155518327 IC50 = 7.42 nM T00612 CCDU61 155518496 IC50 = 205 nM T00612 C5ZQ3R 155519423 IC50 > 1000 nM T00612 CDY5H6 155519645 IC50 = 4910 nM T00612 C34FXY 155520399 IC50 = 9835 nM T00612 CAD10S 155520741 IC50 > 10000 nM T00612 CAZ3S7 155521187 IC50 = 16000 nM T00612 CZ75FW 155521272 IC50 = 203 nM T00612 CG4F2U 155521283 IC50 = 144 nM T00612 C82PHV 155521822 IC50 = 3060 nM T00612 C6DVZ9 155521965 IC50 = 5030 nM T00612 C0KJ1Z 155522601 IC50 > 10000 nM T00612 C63KJW 155523399 IC50 > 1000 nM T00612 CG84WO 155523907 IC50 = 1493 nM T00612 CU5RZ1 155524034 IC50 = 665 nM T00612 CJ3E4G 155524660 IC50 = 6660 nM T00612 CYB97D 155525236 IC50 > 1000 nM T00612 C8DM2Y 155525412 IC50 > 1000 nM T00612 CI24AD 155525662 IC50 = 4214 nM T00612 CN7B1T 155525782 IC50 > 100000 nM T00612 CG1K0O 155526247 IC50 > 10000 nM T00612 COD92I 155526258 IC50 = 3500 nM T00612 C63NOC 155527045 IC50 = 662 nM T00612 CEM0A3 155527290 IC50 = 3222 nM T00612 CW2H5R 155527295 IC50 = 485 nM T00612 C71UNO 155527385 Ki = 70 nM T00612 CQK19H 155527955 IC50 = 786 nM T00612 C20FJM 155528257 IC50 > 1000 nM T00612 CHR4K5 155528532 IC50 > 100000 nM T00612 CZ70PO 155529066 IC50 > 50000 nM T00612 C49NGT 155529137 IC50 > 50000 nM T00612 C9L6OC 155529247 IC50 = 3.4 nM T00612 C94BFW 155529690 IC50 = 5950 nM T00612 C74OTA 155529983 IC50 = 1746 nM T00612 CU0C7W 155530254 IC50 = 500 nM T00612 CZMC49 155530597 IC50 = 24.5 nM T00612 C8AZI6 155530932 IC50 = 7316 nM T00612 CZG79N 155531159 IC50 = 474.1 nM T00612 CN3W5J 155531452 IC50 > 50000 nM T00612 CUC3P1 155531533 IC50 = 1600 nM T00612 CK2UY4 155531957 IC50 > 50000 nM T00612 CDJ0W3 155532052 IC50 = 1080 nM T00612 CZO38U 155532084 IC50 = 1885 nM T00612 CBCJ50 155532192 IC50 > 1000 nM T00612 C3HDI1 155532640 IC50 = 18.49 nM T00612 CD8ZV7 155532950 IC50 = 1820 nM T00612 CIZ46A 155533876 IC50 = 26000 nM T00612 C0T8AS 155533910 IC50 = 926 nM T00612 CPE68B 155534222 IC50 = 7943.28 nM T00612 C4ST9U 155534232 IC50 > 1000 nM T00612 C5FLH0 155535184 IC50 > 1000 nM T00612 C91UNV 155535585 IC50 = 140 nM T00612 C81KIF 155537008 IC50 = 160 nM T00612 C2JH0S 155537112 IC50 = 283 nM T00612 CQV6H0 155537405 IC50 = 8071 nM T00612 C5FRG0 155537455 IC50 = 172 nM T00612 CTF98X 155537473 IC50 = 420 nM T00612 CAG9P4 155537573 IC50 > 50000 nM T00612 C1PFV7 155538765 IC50 = 1817 nM T00612 CLD19W 155539311 IC50 = 1190 nM T00612 CU6V4Q 155539319 IC50 > 50000 nM T00612 CM5UN4 155539714 IC50 = 1366 nM T00612 CBO78Z 155540097 IC50 = 950 nM T00612 C6U0FM 155540189 IC50 = 14000 nM T00612 C6LQT1 155540719 IC50 > 5000 nM T00612 CKN07B 155541358 IC50 = 1267 nM T00612 C7B5NU 155541992 IC50 = 5380 nM T00612 C4T9YC 155542195 IC50 > 100000 nM T00612 CP4L1F 155544459 IC50 = 45000 nM T00612 CNM3P1 155544603 IC50 > 10000 nM T00612 CXR86J 155545078 IC50 > 50000 nM T00612 CCV9J0 155545380 IC50 = 21 nM T00612 C2UN1K 155545446 IC50 = 136 nM T00612 C1JSY3 155545907 IC50 = 135 nM T00612 C8DQ7U 155546022 IC50 = 107.5 nM T00612 CE1D7Q 155546207 IC50 > 100000 nM T00612 CF2O4J 155546325 IC50 > 50000 nM T00612 CK45LA 155546486 IC50 = 7943.28 nM T00612 C3HB0U 155546555 IC50 = 1995.26 nM T00612 CS3GO2 155546558 IC50 = 850 nM T00612 C0AU1L 155546632 IC50 > 50000 nM T00612 C8LT4A 155546691 IC50 = 67.48 nM T00612 CP3Q7I 155547009 IC50 = 8100 nM T00612 CHD0I6 155547367 IC50 = 2440 nM T00612 C1D4PI 155547606 Ki = 150 nM T00612 CTFU61 155549051 IC50 = 610 nM T00612 C90FBZ 155549087 IC50 > 50000 nM T00612 CE0YL6 155549538 IC50 = 200 nM T00612 CO6ID4 155550122 IC50 = 1000 nM T00612 CV4QP6 155550492 IC50 > 1000 nM T00612 C4Z5JX 155550827 IC50 = 50000 nM T00612 CA03BO 155551057 IC50 = 3162.28 nM T00612 C3JQ1N 155551780 IC50 = 668 nM T00612 C05ZVG 155552130 IC50 = 8320 nM T00612 CV4Y5B 155552792 IC50 = 1100 nM T00612 CXT8F1 155552802 IC50 = 12930 nM T00612 CH8L1V 155554197 IC50 = 860 nM T00612 CGDF76 155554360 IC50 = 24000 nM T00612 CC56ED 155554844 IC50 = 21 nM T00612 CXGR50 155555191 IC50 = 880 nM T00612 C8ZD2Y 155555330 IC50 = 4200 nM T00612 CF2H3O 155555451 IC50 = 489 nM T00612 CM7FN8 155555499 IC50 = 160 nM T00612 CFW90N 155555562 IC50 = 1.6 nM T00612 C8FZN4 155555652 IC50 > 1000 nM T00612 C7QTU1 155555957 IC50 > 50000 nM T00612 CIN57Q 155556138 IC50 = 1130 nM T00612 C6IL1E 155557199 IC50 = 278.6 nM T00612 CEX5I7 155557262 IC50 > 1000 nM T00612 CNM71L 155557418 IC50 = 579.3 nM T00612 C8AUB0 155558567 IC50 = 75 nM T00612 CK3B2T 155558642 IC50 = 3700 nM T00612 CPD50Q 155559583 IC50 = 3400 nM T00612 C26QOJ 155559606 IC50 > 1000 nM T00612 CC62UI 155559872 IC50 = 1810 nM T00612 CT31YW 155560779 IC50 = 7000 nM T00612 C13TBU 155560878 IC50 > 1000 nM T00612 CW50YA 155561265 IC50 = 1298 nM T00612 CH0Z1P 155561539 IC50 = 352 nM T00612 CJ4KO7 155562145 IC50 = 441.3 nM T00612 CGL24S 155562249 IC50 > 50000 nM T00612 CSJ23C 155562809 IC50 = 994 nM T00612 CM0DS1 155562992 IC50 > 1000 nM T00612 CBJ03Y 155563284 IC50 = 819 nM T00612 CXEQ27 155563524 IC50 = 1400 nM T00612 CXWU93 155563558 IC50 = 180 nM T00612 CX23YB 155564400 IC50 = 95.51 nM T00612 CR85ZW 155564587 IC50 = 1900 nM T00612 CPNA06 155564750 IC50 > 50000 nM T00612 C87JXN 155564870 IC50 = 6309.57 nM T00612 CG65CR 155565674 IC50 = 50000 nM T00612 CD05RS 155566122 IC50 > 50000 nM T00612 C4A0RK 155566461 IC50 > 50000 nM T00612 CP1MH4 155566833 IC50 = 8300 nM T00612 C04CGS 155567444 IC50 > 50000 nM T00612 CDT3W1 155567506 IC50 > 1000 nM T00612 CS03PJ 155568350 IC50 > 50000 nM T00612 CF2X0U 155568767 IC50 = 530 nM T00612 CW5XB4 155569484 IC50 = 147 nM T00612 C3BAZ5 24861442 IC50 = 12.7 nM T00612 D00GBB 11449246 Ki = 44 nM T00612 D00HXX 56650312 IC50 = 9700 nM T00612 D00KFF 9882812 IC50 = 1400 nM T00612 D00SEE 11379392 IC50 = 1300 nM T00612 D01AVS 25065930 IC50 = 500 nM T00612 D01FYB 23648267 IC50 = 2000 nM T00612 D01TSM 46887380 IC50 = 3800 nM T00612 D01YBR 44591988 IC50 = 27700 nM T00612 D02NWS 279980 Ki = 430 nM T00612 D02TQA 15986508 IC50 = 1860 nM T00612 D03QOD 239512 IC50 = 6600 nM T00612 D03TNE 25065710 IC50 = 500 nM T00612 D03TQD 25065713 IC50 = 500 nM T00612 D04KQF 6675804 Ki = 42 nM T00612 D04UVL 1133083 IC50 = 6980 nM T00612 D05OVV 11993691 IC50 = 2000 nM T00612 D05RWU 46887334 IC50 = 800 nM T00612 D06IWR 46887438 IC50 = 1300 nM T00612 D07BMT 46887378 IC50 = 3900 nM T00612 D07MYE 5355635 IC50 = 457 nM T00612 D07WSB 46887381 IC50 = 3100 nM T00612 D07YZZ 5173 Ki = 29 nM T00612 D08USK 46887437 IC50 = 13000 nM T00612 D08YLO 46830345 IC50 = 1400 nM T00612 D09RKA 72946782 IC50 = 0.112 nM T00612 D09SVH 25065929 IC50 = 500 nM T00612 D0A4KW 46830327 IC50 = 39 nM T00612 D0AK8Q 42632368 IC50 = 820 nM T00612 D0B3ZM 11436024 IC50 = 2220 nM T00612 D0D2US 25065931 IC50 = 500 nM T00612 D0E0TA 44454650 IC50 = 200 nM T00612 D0E9DD 16095101 Ki = 50 nM T00612 D0FI2F 25065925 IC50 = 500 nM T00612 D0G6DH 16661454 IC50 = 870 nM T00612 D0H4SC 46887439 IC50 = 600 nM T00612 D0H4YW 3611 Ki = 15.44 nM T00612 D0I2KC 46830328 IC50 = 43 nM T00612 D0K3MR 22915475 IC50 = 720 nM T00612 D0K7QR 45269423 IC50 = 590 nM T00612 D0M1ZI 16095112 Ki = 3000 nM T00612 D0M9LJ 44454415 IC50 = 900 nM T00612 D0MD7H 44454143 IC50 = 27 nM T00612 D0N9AK 44138031 IC50 = 11000 nM T00612 D0Q2GM 44454416 IC50 = 390 nM T00612 D0Q4LX 46887475 IC50 = 10000 nM T00612 D0Q5DI 71462653 Ki = 1250 nM T00612 D0Q5MC 24753719 IC50 = 31000 nM T00612 D0Q9PO 16095114 Ki = 10 nM T00612 D0T0SK 44138032 IC50 = 2670 nM T00612 D0T4JQ 264 IC50 = 12000 nM T00612 D0U8FC 759408 IC50 = 3100 nM T00612 D0W1PV 6918328 Ki = 0.12 nM T00612 D0W2PX 46887379 IC50 = 140 nM T00612 D0W9BH 15986510 IC50 = 330 nM T00612 D0X4VO 44359538 IC50 = 26000 nM T00612 D0XZ9Q 11149404 IC50 = 754 nM T00612 D0Y4SD 46887333 IC50 = 390 nM T00612 D0YO6M 785232 IC50 = 900 nM T00612 D0Z8PX 24757913 IC50 = 18.65 nM T89772 CZ6G7B 69873 IC50 = 90000 nM T89772 CU0HZ5 148839 IC50 = 2000 nM T89772 CGV04U 264832 IC50 = 10000 nM T89772 C06KJA 369967 Ki = 170 nM T89772 C6P0NL 369973 Ki = 30 nM T89772 CQFU62 449639 Ki = 0.44 nM T89772 C35WDY 659840 Ki = 2 nM T89772 CAHN76 833992 IC50 = 500 nM T89772 CTQS24 3078235 IC50 = 300 nM T89772 CH60OS 3078239 IC50 = 10 nM T89772 CH16JM 3083476 Ki = 0.36 nM T89772 CKPD73 9859994 Ki = 2900 nM T89772 CKMW59 9957260 Ki = 0.3 nM T89772 C9DJ0L 9982983 Ki = 0.45 nM T89772 C6WY0U 9999116 Ki = 0.22 nM T89772 CU18XB 10069224 Ki = 0.36 nM T89772 C5T7DN 10316732 IC50 = 34 nM T89772 CGT74I 10317813 Ki = 10.7 nM T89772 C4K9SA 10334147 Ki = 7.6 nM T89772 C4QN0C 10385293 Ki = 0.77 nM T89772 CN62ZX 10436105 Ki = 0.67 nM T89772 CJRB30 10567286 Ki = 0.44 nM T89772 CY9O0S 10573578 Ki = 33 nM T89772 CGJ0K6 10618918 Ki = 570 nM T89772 CL8E5M 10717134 Ki = 0.99 nM T89772 C35BVU 10717135 Ki = 10 nM T89772 CKTU76 10744775 Ki = 5.2 nM T89772 C3EK9S 10768549 Ki = 0.26 nM T89772 CN6CQ0 10780604 Ki = 74 nM T89772 C1OYW8 10807685 Ki = 77 nM T89772 CX6U3K 10807863 Ki = 85 nM T89772 C2TPA5 10814571 Ki = 0.4 nM T89772 CB60JU 11546462 IC50 = 11 nM T89772 C4X8UL 11800052 Ki = 17 nM T89772 CP06IE 13119693 IC50 > 40000 nM T89772 CW4S8E 13816598 IC50 = 10000 nM T89772 CU0BJ4 15925754 IC50 = 200 nM T89772 CO4Q7Y 15925755 IC50 = 200 nM T89772 C1BHO7 15925759 IC50 = 40000 nM T89772 C6TOS0 15925762 IC50 = 40 nM T89772 C7DJ0E 15925764 IC50 = 100 nM T89772 C7A2RX 15925766 IC50 = 300 nM T89772 CCZ0K7 15925767 IC50 = 70 nM T89772 C7JVN5 15925769 IC50 = 1000 nM T89772 CAVF72 15925771 IC50 = 50 nM T89772 CZL8B3 15925773 IC50 = 5000 nM T89772 CH8B3Y 15925776 IC50 = 3000 nM T89772 C02UIF 15925779 IC50 = 4000 nM T89772 C2DBF5 15925781 IC50 = 20000 nM T89772 C6IQ2G 15925786 IC50 = 500 nM T89772 C8FRY1 15925788 IC50 = 300 nM T89772 C10LJQ 15925790 IC50 = 300 nM T89772 C2BM6N 15925792 IC50 > 1000 nM T89772 C9GJ4Q 15925794 IC50 = 200 nM T89772 CSZA10 15925796 IC50 = 1000 nM T89772 CSN08P 15925798 IC50 = 2000 nM T89772 CB02FC 15925801 IC50 = 20 nM T89772 CRO8K2 15925804 IC50 = 90 nM T89772 C6T9JV 15925806 IC50 = 600 nM T89772 CO3C0G 15925810 IC50 = 200 nM T89772 C2DQI0 15925812 IC50 = 200 nM T89772 C8XO9R 15925813 IC50 = 100 nM T89772 C7HN9X 15925815 IC50 = 300 nM T89772 CJB1E9 15925818 IC50 = 100 nM T89772 C6IXC7 15925820 IC50 = 500 nM T89772 CM8K0C 15925822 IC50 = 20000 nM T89772 C6R4TF 15925824 IC50 = 300 nM T89772 C3QS2V 15925826 IC50 = 400 nM T89772 CH61AK 15925830 IC50 = 300 nM T89772 C8J2IL 15925832 IC50 = 2000 nM T89772 C4UD7M 15925834 IC50 = 2000 nM T89772 CB3P0Z 15925838 IC50 > 1000 nM T89772 C7Q0PV 15925842 IC50 = 2000 nM T89772 CYX92F 15925844 IC50 = 8000 nM T89772 C0R1BG 15925846 IC50 = 5000 nM T89772 C7XDG6 15925854 IC50 = 300 nM T89772 CDRY47 15925856 IC50 = 100 nM T89772 C1WV0Y 15925857 IC50 > 2000 nM T89772 CDN6B8 15925859 IC50 = 50 nM T89772 CK3OT2 15925860 IC50 = 300 nM T89772 CJFU26 15925862 IC50 = 50 nM T89772 CM8D1I 15925864 IC50 = 500 nM T89772 CRJ3T9 15925866 IC50 = 100 nM T89772 CLS1I9 15925870 IC50 = 1000 nM T89772 CJP40F 15925875 IC50 = 200 nM T89772 CEM0C4 15925877 IC50 = 300 nM T89772 CN12QC 15925880 IC50 = 20000 nM T89772 C4FAB0 15925883 IC50 = 40000 nM T89772 CV31EJ 15925885 IC50 = 10000 nM T89772 CAB58D 15925887 IC50 = 100 nM T89772 C1DQ9F 15925889 IC50 = 800 nM T89772 CHG68S 15925891 IC50 = 9000 nM T89772 C5ACX2 15925894 IC50 = 4000 nM T89772 C37RKM 15925895 IC50 = 4000 nM T89772 C1C2DX 15925897 IC50 = 1000 nM T89772 C89BVA 15925900 IC50 = 100 nM T89772 C4XHY1 15925902 IC50 = 800 nM T89772 C54EHD 15925903 IC50 = 3000 nM T89772 CPYG78 15925906 IC50 = 3000 nM T89772 C64SNC 15925909 IC50 = 10000 nM T89772 C16HSM 15925911 IC50 = 300 nM T89772 C32RJT 15925916 IC50 = 50 nM T89772 C3EMR4 15925918 Ki = 0.055 nM T89772 CDMT40 15925919 IC50 = 100 nM T89772 CG4HF5 15925921 IC50 = 2000 nM T89772 CHGU25 15925923 IC50 = 80000 nM T89772 CL8Y9M 15925925 IC50 > 100000 nM T89772 C2S4ED 25233584 Ki = 0.25 nM T89772 C2WT7K 25233585 Ki = 1.68 nM T89772 C9N8CT 25233586 Ki = 2.7 nM T89772 C7BC2Z 25233762 Ki = 4.3 nM T89772 CFGZ21 25233763 Ki = 0.48 nM T89772 C8M5WY 44274109 IC50 = 6000 nM T89772 CYP17T 44350537 Ki = 144 nM T89772 CD38RO 44350538 Ki = 298 nM T89772 C0K5CR 44350649 Ki = 130 nM T89772 CCU89V 44350664 Ki = 594 nM T89772 C3JAW4 44350676 Ki = 380.11 nM T89772 C3CM2E 44350704 Ki = 3400 nM T89772 C03YVC 44350708 Ki = 60 nM T89772 CC3Y4A 44350710 Ki = 411 nM T89772 C8EF0H 44350786 Ki = 474 nM T89772 C5E3FK 44350787 Ki = 182 nM T89772 C41UID 44350800 Ki = 14.5 nM T89772 CRC5I3 44350810 Ki = 325 nM T89772 C69MTC 44350812 Ki = 420 nM T89772 CMRX47 44350817 Ki = 8.5 nM T89772 CZMW86 44350827 Ki = 10.3 nM T89772 CI7KH4 44350870 Ki = 8.5 nM T89772 C7NC0V 44350885 Ki = 600 nM T89772 C60IJH 44350886 Ki = 86 nM T89772 CPF13Q 44410771 IC50 = 66 nM T89772 CY85XC 44410772 IC50 > 100 nM T89772 CS3M6N 44410774 IC50 > 100 nM T89772 CRC6X0 44410775 IC50 > 100 nM T89772 CJ2Z9N 44410776 IC50 > 100 nM T89772 CLG2T9 44410778 IC50 > 100 nM T89772 C2C7FK 44410785 IC50 > 100 nM T89772 CQ4F1N 44410786 IC50 > 1000 nM T89772 C71CMX 44410787 IC50 > 100 nM T89772 C2CI3R 44410788 IC50 > 100 nM T89772 C6TBH7 44410813 IC50 > 1000 nM T89772 CIR06J 44410883 IC50 = 100 nM T89772 CXWH78 44410884 IC50 = 57 nM T89772 C5O3WP 44410885 IC50 > 100 nM T89772 CVX4T1 44410886 IC50 > 100 nM T89772 CKI08N 44410890 IC50 = 47 nM T89772 COM35A 44410891 IC50 = 46 nM T89772 C0DZT7 44410897 IC50 > 100 nM T89772 CWA19Z 44410919 IC50 = 100 nM T89772 CBX46M 44410922 IC50 > 1000 nM T89772 CF9AM3 44410923 IC50 > 100 nM T89772 C0N2XB 44474938 Ki > 1 nM T89772 CF4GY9 44564272 Ki = 330 nM T89772 C0R6OL 46197218 Ki = 5 nM T89772 CU63SQ 50994498 Ki = 1.4 nM T89772 CEIG81 53391632 Ki = 1360 nM T89772 CIU6Z7 53391633 Ki = 3310 nM T89772 CC8XY3 53391634 Ki = 401 nM T89772 CLNG65 53391635 Ki = 2030 nM T89772 CQ3M2A 53391731 Ki = 294 nM T89772 C17KBN 53391732 Ki = 14800 nM T89772 CT76BC 53391733 Ki = 44.2 nM T89772 CR49GI 53391734 Ki = 137 nM T89772 CHSU87 53391735 Ki = 3600 nM T89772 CN4W7D 53391736 Ki = 30900 nM T89772 CRBY03 53391833 Ki = 683 nM T89772 C6OTS5 53391834 Ki = 3340 nM T89772 C3Q7GW 53391835 Ki = 3460 nM T89772 C23ZDG 53391836 Ki = 555 nM T89772 CGQ71S 53391837 Ki = 372 nM T89772 CSEX93 53391838 Ki = 136 nM T89772 C1W8RI 53391950 Ki = 1970 nM T89772 CXY8S2 53391951 Ki = 149 nM T89772 CC7K8L 53391952 Ki = 237 nM T89772 CMA3R8 53391953 Ki = 48.6 nM T89772 CR7S4M 53391954 Ki = 1080 nM T89772 CA8QX4 53391955 Ki = 35.5 nM T89772 CFR8Z9 53392068 Ki = 107 nM T89772 C7WT2D 54290606 IC50 = 2000 nM T89772 CG67HW 56678898 Ki = 22.9 nM T89772 CUL3W2 57402462 Ki > 1 nM T89772 C5AC7T 70641778 Ki = 19 nM T89772 C3VIW7 70681946 Ki = 1190 nM T89772 CMW81Z 70684064 Ki = 8700 nM T89772 C7SU3Q 70684070 Ki = 15.4 nM T89772 C7KF2Z 70684072 Ki = 206 nM T89772 C57JFX 70686208 Ki = 810 nM T89772 CQP0C7 70686210 Ki = 123 nM T89772 C1KLY9 70686215 Ki = 142 nM T89772 C2T0WU 70690343 Ki = 13000 nM T89772 C7MX1S 70690345 Ki = 3020 nM T89772 C5IEG9 70690354 Ki = 19 nM T89772 CUQT52 70690356 Ki = 10.2 nM T89772 CN6HB7 70691042 IC50 = 1000 nM T89772 C9JXG2 70694568 Ki = 112 nM T89772 CTGU74 70694570 Ki = 2020 nM T89772 CX53BM 70694572 Ki = 1350 nM T89772 CQ5C1W 70696607 Ki = 62.7 nM T89772 C35TZP 70696609 Ki = 11.4 nM T89772 CA1ZO2 70696611 Ki = 233 nM T89772 C6B8MO 70696616 Ki = 1300 nM T89772 C1KH6U 71719166 Ki = 211 nM T89772 CAB02F 73346026 Ki = 3.03 nM T89772 C5XMI8 73347556 Ki = 38 nM T89772 C2R4LO 73347557 Ki = 23.3 nM T89772 C59NZD 73347558 Ki = 8.36 nM T89772 C68HNS 73347559 Ki = 121 nM T89772 C4F7YE 73349091 Ki = 48 nM T89772 CH5M9F 73349092 Ki = 2310 nM T89772 CKY9Z2 73350664 Ki = 0.93 nM T89772 C80WEF 73350665 Ki = 38.7 nM T89772 C86WNX 73350666 Ki = 18.4 nM T89772 COG43D 73352164 Ki = 118 nM T89772 CWP0I6 73352165 Ki = 27.9 nM T89772 CU2JG9 73353623 Ki = 26.1 nM T89772 CZOM24 73355118 Ki = 12.7 nM T89772 CHVZ43 73355119 Ki = 24.1 nM T89772 CX0KB4 73356685 Ki = 10.1 nM T89772 CB42TQ 73356686 Ki = 66.2 nM T89772 C3SZC9 73356687 Ki = 182 nM T89772 CS3Q2K 73356688 Ki = 76.4 nM T89772 C2LD9V 73356689 Ki = 26.6 nM T89772 C0IH5W 122183457 Ki = 1.74 nM T89772 CR7S9G 122183458 Ki = 0.87 nM T89772 CGVW94 122183459 Ki = 1.23 nM T89772 CO3JF1 122183460 Ki = 4.64 nM T89772 C7G1VF 122183461 Ki = 56.2 nM T89772 C1H6WO 122183462 Ki = 1.55 nM T89772 C5ZBJ6 122183463 Ki = 0.59 nM T89772 C9JG3P 122183464 Ki = 92.8 nM T89772 C5SLG8 122183466 Ki = 2.7 nM T89772 CWF82K 450854 Ki = 0.32 nM T89772 CN1DM0 57402731 Ki = 27.5 nM T89772 C8NBM0 71817329 Ki = 0.78 nM T89772 D0I1QF 5662 IC50 = 40 nM T89772 D0JB1D 9399 IC50 = 12 nM T89772 D0N8WR 10390222 Ki = 0.13 nM T20891 D03MNN 11341869 IC50 > 1000 nM T20891 D03RTS 2662 IC50 = 48000 nM T20891 D0J9ZR 4477 IC50 = 83900 nM T20891 D02RJY 11442891 IC50 > 10000 nM T20891 D07EHV 44814409 IC50 > 10000 nM T20891 D07HPJ 11476171 IC50 = 8900 nM T20891 D0C9JJ 10027278 IC50 = 5000 nM T20891 D0E3TC 44259 IC50 = 10 nM T20891 D0M0XB 10302451 IC50 > 10000 nM T20891 D0O0LS 25141092 IC50 > 10000 nM T20891 D0Q9UX 16718576 IC50 > 10000 nM T20891 D0W3LI 153999 IC50 = 750 nM T20891 D0YK9D 9956119 IC50 > 10000 nM T20891 D0ZE5U 11161844 IC50 = 5 nM T20891 D0L5YF 5329032 IC50 > 20000 nM T20891 CKJH62 13399 IC50 = 311000 nM T20891 C0C5AB 24057 IC50 = 256000 nM T20891 CZJ8U9 30976 IC50 = 50800 nM T20891 CM0Q2H 70632 IC50 = 340000 nM T20891 C56RJL 88336 IC50 = 160000 nM T20891 C7WS2Q 150896 IC50 = 169000 nM T20891 C12ODI 221158 IC50 = 90800 nM T20891 CJ0T9Y 311869 IC50 = 376000 nM T20891 C2NX8S 403053 IC50 = 828000 nM T20891 C1ZG2U 449087 IC50 > 10000 nM T20891 C5UM8B 513197 IC50 = 58700 nM T20891 CDG5N8 523183 IC50 = 313000 nM T20891 C51ERD 547494 IC50 = 95100 nM T20891 CYG1F2 580973 IC50 = 200000 nM T20891 CQ59SY 639665 IC50 = 6600 nM T20891 CW12BK 657138 IC50 = 39 nM T20891 C65QBR 794624 IC50 = 60000 nM T20891 CZJB27 817910 IC50 = 101900 nM T20891 C6D4RC 845961 IC50 = 61000 nM T20891 CB57ZE 969430 IC50 = 402000 nM T20891 C9NJ1L 1858265 IC50 = 200 nM T20891 CJ1MA7 2728593 EC50 = 133000 nM T20891 CWCH42 2786631 IC50 = 82400 nM T20891 C7DNX2 2849295 EC50 = 2000 nM T20891 CA9OH8 4057787 IC50 = 29000 nM T20891 C5SY4O 5330420 IC50 > 10 nM T20891 CGAT56 5494442 IC50 = 200 nM T20891 CM5Z8X 9869943 IC50 > 1000 nM T20891 CJO47T 9948405 IC50 > 10000 nM T20891 CV8I5X 9999342 IC50 > 10000 nM T20891 CINF40 10073694 IC50 = 570 nM T20891 C5TQ7X 10247543 IC50 > 10000 nM T20891 C8RD3V 10301884 IC50 > 10000 nM T20891 C32SGV 10343467 IC50 = 2000 nM T20891 C0IVL9 10347359 IC50 = 2.3 nM T20891 CVN8T9 10379252 IC50 = 1100 nM T20891 C2B0IU 10421236 IC50 = 5400 nM T20891 C2WQ8M 10473563 IC50 > 10000 nM T20891 CAZT53 10475366 IC50 > 25000 nM T20891 CJWH60 10489322 IC50 = 510 nM T20891 CO2DA6 11165945 IC50 = 1000 nM T20891 C8Y6IM 11234514 IC50 = 34 nM T20891 C3T6XF 11256709 IC50 = 1000 nM T20891 CBOP58 11293798 Ki = 2070 nM T20891 CN0VA4 11323104 IC50 = 55 nM T20891 C8XIF5 11350077 IC50 = 110 nM T20891 C26BZX 11362471 Ki = 740 nM T20891 COF6V0 11370369 IC50 > 10000 nM T20891 C5EP3S 11373564 IC50 = 1000 nM T20891 CWXB93 11397177 Ki > 10000 nM T20891 C4OT0X 11417334 IC50 = 1000 nM T20891 C0APW4 11422034 IC50 > 10000 nM T20891 CW53GT 11440050 IC50 > 10000 nM T20891 C93UPX 11447681 IC50 = 990 nM T20891 C5H7KT 11453730 IC50 = 1000 nM T20891 C67RAF 11461275 IC50 = 14 nM T20891 C0KLW5 11514099 IC50 = 21200 nM T20891 CAP6N0 11588244 IC50 = 100 nM T20891 C68RNE 11738018 IC50 = 3 nM T20891 CY8C9P 11751126 IC50 > 25000 nM T20891 CHD8K3 11774303 IC50 = 327 nM T20891 CDZ1I3 11989153 IC50 = 340 nM T20891 C2RQ1E 12508473 IC50 = 344000 nM T20891 CETK42 12628603 IC50 = 102000 nM T20891 CAI5N8 13415516 IC50 = 97500 nM T20891 CFPW41 16007116 Ki > 3800 nM T20891 C9TU1O 16046126 IC50 > 1000 nM T20891 C2LA8B 16412755 IC50 = 326000 nM T20891 C2IF3P 16678352 IC50 = 11200 nM T20891 C3IO1C 16679060 IC50 > 30000 nM T20891 C0TMW8 16739778 IC50 = 1400 nM T20891 CJE01Z 16956491 IC50 = 273000 nM T20891 CM4OH5 17028040 EC50 = 40000 nM T20891 CVS0T5 17754396 IC50 = 60 nM T20891 CP01IJ 17754397 IC50 = 270 nM T20891 C48WLO 17754398 IC50 = 580 nM T20891 C4TZP6 17754449 IC50 = 2120 nM T20891 CNQX79 17754450 IC50 = 40 nM T20891 C5GA2P 17754539 IC50 = 60 nM T20891 CZ3UJ5 17754582 IC50 = 200 nM T20891 CC2VO6 17754723 IC50 = 670 nM T20891 C0HE8A 17754724 IC50 = 7450 nM T20891 CJ5X6R 17754761 IC50 = 260 nM T20891 CW6A3F 20289271 IC50 = 244000 nM T20891 C0X3KJ 21051556 IC50 = 67 nM T20891 CXLN26 21957724 IC50 = 3900 nM T20891 CO3JZ1 21957734 IC50 > 26000 nM T20891 CW8UV9 21957747 IC50 > 26000 nM T20891 CPH76G 21957770 IC50 = 4200 nM T20891 CM7N4G 21957818 IC50 = 10 nM T20891 C2F0GM 22319690 IC50 = 13200 nM T20891 C9QLP0 23133323 IC50 > 20000 nM T20891 C5Y1QX 23644715 IC50 = 260 nM T20891 CY8Z7X 23647330 IC50 > 10000 nM T20891 C4XD8H 23647348 IC50 > 10000 nM T20891 CWE47K 23647595 IC50 > 10000 nM T20891 CICB91 23647596 IC50 = 100 nM T20891 C7W0PE 23647597 IC50 = 1000 nM T20891 CTI1F7 23647598 IC50 = 20 nM T20891 CSOG98 23647599 IC50 = 10 nM T20891 CUX5O6 23647602 IC50 > 1000 nM T20891 CA4LE6 23647603 IC50 = 1000 nM T20891 CX3H1O 23647607 IC50 = 2700 nM T20891 CM3G9W 23647608 IC50 = 1000 nM T20891 CEUR56 23647609 IC50 = 900 nM T20891 C4G3IX 23647610 IC50 = 80 nM T20891 CP4HE0 23647611 IC50 = 280 nM T20891 C17FBN 23647612 IC50 = 280 nM T20891 CAF1V6 23647613 IC50 = 680 nM T20891 C4DO5F 23647614 IC50 = 2300 nM T20891 C9KQX5 23647615 IC50 = 580 nM T20891 C6OS7T 23647616 IC50 = 290 nM T20891 CGD7R2 23647617 IC50 = 670 nM T20891 CSYB42 23647618 IC50 = 120 nM T20891 CBD9U4 23647620 IC50 = 580 nM T20891 C0SFX2 23647621 IC50 = 1000 nM T20891 C6E1PQ 23647622 IC50 = 530 nM T20891 CEYZ50 23647623 IC50 = 29 nM T20891 CEP8V7 23647624 IC50 = 34 nM T20891 C48ZIV 23647625 IC50 = 6100 nM T20891 CJK9L4 23647626 IC50 = 5400 nM T20891 CBDU83 23647627 IC50 = 9 nM T20891 CRUB96 23648180 IC50 = 290 nM T20891 CK8QI1 23648181 IC50 = 970 nM T20891 C0A9EN 23648219 IC50 = 2490 nM T20891 CH2JK3 24729254 IC50 = 163600 nM T20891 C7YG1N 24759534 IC50 = 130 nM T20891 CCP2M3 24822704 IC50 > 50000 nM T20891 C4YPL5 24860827 IC50 > 10000 nM T20891 CSY5F8 25059884 IC50 = 1864 nM T20891 C2Q8EV 25059887 IC50 = 7490 nM T20891 CXLR35 25060138 IC50 = 2064 nM T20891 CG7WZ4 25060408 IC50 = 43 nM T20891 CL7V8R 25060409 IC50 = 3 nM T20891 CFU5E2 25060410 IC50 = 6 nM T20891 C3B8FI 25060411 IC50 = 8 nM T20891 C4CJX9 25060675 IC50 = 21 nM T20891 CLP07J 25110819 IC50 = 1100 nM T20891 CLP92Q 25164369 IC50 = 1200 nM T20891 C32ALZ 25164370 IC50 = 2200 nM T20891 C8MFK3 25164571 IC50 = 390 nM T20891 C0E2DP 25164572 IC50 = 1000 nM T20891 C30XCK 25164971 IC50 = 480 nM T20891 CQ0VN5 25164974 IC50 > 10000 nM T20891 CNC30U 25165168 IC50 > 10000 nM T20891 C4LHV1 25165368 IC50 = 85 nM T20891 C1LM6S 25165369 IC50 = 500 nM T20891 CHXD34 25165370 IC50 = 450 nM T20891 C2CXH3 25165371 IC50 = 170 nM T20891 CQWL59 25165372 IC50 = 28000 nM T20891 CTY05L 25165575 IC50 = 3500 nM T20891 CL87JW 25165773 IC50 = 13 nM T20891 CB89TL 25165774 IC50 = 260 nM T20891 CZH3Q1 25165775 IC50 = 2400 nM T20891 CB0NZ6 25165959 IC50 = 2700 nM T20891 CFZI92 25165961 IC50 = 110 nM T20891 CVI75Q 25167375 IC50 = 1800 nM T20891 CH73US 25628008 EC50 = 50000 nM T20891 CC71QJ 27666048 IC50 > 100000 nM T20891 C2UZ0E 44176356 IC50 = 70 nM T20891 CU19EF 44231127 IC50 = 580 nM T20891 C53BSX 44236913 IC50 = 739 nM T20891 C73PKN 44236914 IC50 = 108 nM T20891 CTL61O 44236915 IC50 = 2033 nM T20891 CK9JF1 44236916 IC50 = 100 nM T20891 C64SRV 44236917 IC50 > 1000 nM T20891 C4DXL0 44236918 IC50 = 66 nM T20891 C2V5AG 44236919 IC50 > 100 nM T20891 C0Y6NR 44236920 IC50 = 6923 nM T20891 CK0T6S 44236921 IC50 = 35 nM T20891 C92AOQ 44236922 IC50 = 74 nM T20891 CODK43 44236923 IC50 = 146 nM T20891 CVNB79 44236924 IC50 = 144 nM T20891 CPN70A 44236925 IC50 = 26 nM T20891 C1F9YM 44236926 IC50 = 57 nM T20891 CXZ8V7 44236927 IC50 = 65 nM T20891 C0W9KP 44236928 IC50 = 532 nM T20891 CZ3F6E 44236929 IC50 > 1000 nM T20891 C93QWS 44236930 IC50 = 283 nM T20891 CJ70YM 44236931 IC50 = 74 nM T20891 C86XBN 44236932 IC50 = 434 nM T20891 CC92ET 44236933 IC50 = 383 nM T20891 C9O7AR 44236934 IC50 = 47 nM T20891 CGZ0X8 44236935 IC50 = 67 nM T20891 CO17JA 44236936 IC50 = 142 nM T20891 CGN1T9 44236937 IC50 = 24 nM T20891 C3H1OQ 44236938 IC50 = 91 nM T20891 CWR81Q 44236939 IC50 = 51 nM T20891 C97ENG 44236940 IC50 = 30 nM T20891 C4FH9P 44236941 IC50 = 505 nM T20891 CC72GH 44236942 IC50 > 1000 nM T20891 CV3KY6 44434101 IC50 = 300 nM T20891 CO9U0G 44434107 IC50 = 1180 nM T20891 CC7O6L 44454395 IC50 = 150 nM T20891 C9ZML1 44454396 IC50 = 245 nM T20891 C3VRO9 44557921 IC50 > 10000 nM T20891 CHKQ45 44593990 IC50 = 58 nM T20891 CY3SV7 44596118 IC50 = 82 nM T20891 CVW08Q 44608012 IC50 = 8 nM T20891 C1SIK2 44620952 IC50 = 17 nM T20891 CES64N 45139232 Ki = 100 nM T20891 C0U1IR 45139233 Ki = 0.6 nM T20891 CK49WN 45139234 Ki = 1.4 nM T20891 C8J5VB 45381792 EC50 = 60000 nM T20891 CQYO76 46192856 IC50 = 5 nM T20891 CU1Q0K 46192857 IC50 = 6 nM T20891 CQ82JV 46192858 IC50 = 3 nM T20891 CN0A1I 46192859 IC50 = 14 nM T20891 CM96WL 46192860 IC50 = 18 nM T20891 CDJS49 46192989 IC50 = 3 nM T20891 CS9T2M 46192991 IC50 = 15 nM T20891 CD4O0S 46192992 IC50 = 13 nM T20891 CPK5N7 46193129 IC50 = 6 nM T20891 CQ8YW5 46193130 IC50 = 15 nM T20891 C3VYA4 46193131 IC50 = 8 nM T20891 CS5Q2R 46193132 IC50 = 6 nM T20891 C52HOD 46193133 IC50 = 9 nM T20891 C8ADR2 46214481 IC50 = 199.53 nM T20891 CH0ZR1 46214482 IC50 = 125.89 nM T20891 C2EZU8 46214649 IC50 = 50.12 nM T20891 C5L1KH 46214650 IC50 = 251.19 nM T20891 CRI6G5 46214652 IC50 = 158.49 nM T20891 CRT51W 46214653 IC50 = 316.23 nM T20891 CVW21C 46215644 IC50 = 19.95 nM T20891 CZ58FY 46215814 IC50 = 370 nM T20891 CO9H1K 46215816 IC50 = 655 nM T20891 CT8G2A 46215988 IC50 = 63.1 nM T20891 C28SJK 46215992 IC50 = 31.62 nM T20891 C9JNT0 46216155 IC50 = 5.012 nM T20891 CD96WF 46216494 IC50 = 251.19 nM T20891 CY3HW5 46224684 IC50 = 53 nM T20891 CYV1U4 46829289 IC50 = 374 nM T20891 CLS29B 46872626 IC50 > 10000 nM T20891 C3T0VS 46911003 IC50 = 85 nM T20891 CFE24L 46911770 IC50 = 36 nM T20891 C19JYF 49766501 EC50 = 1 nM T20891 CWU7F5 49798058 IC50 = 2740 nM T20891 CJ3R5V 49798446 EC50 = 900000 nM T20891 CNYT10 49798471 EC50 = 101000 nM T20891 C8A2DC 49798539 EC50 = 23000 nM T20891 C9L1SQ 49798540 EC50 = 53000 nM T20891 CC4QU2 49798541 EC50 = 187000 nM T20891 C0CSZ8 49798542 EC50 = 75000 nM T20891 C01EXF 49798577 EC50 = 45000 nM T20891 CHSF07 49806372 IC50 > 1000 nM T20891 CF91RS 49843531 IC50 > 10000 nM T20891 CMX95S 49863380 EC50 = 14200 nM T20891 CRCT70 50909914 IC50 = 19.95 nM T20891 C0XDI4 50909915 IC50 = 333 nM T20891 CUJL92 50909916 IC50 = 10 nM T20891 C51DKX 50909917 IC50 = 74 nM T20891 C2Y6QS 50938552 IC50 > 10000 nM T20891 C9NYP4 51036677 IC50 > 10000 nM T20891 C4WRY3 51037112 IC50 > 10000 nM T20891 CRI28Z 51037948 IC50 > 10000 nM T20891 CYD4A2 51354035 IC50 = 3.162 nM T20891 CW2T3N 51354036 IC50 = 3.162 nM T20891 CH8NX6 51354037 IC50 = 6.31 nM T20891 CK63DI 51354327 IC50 = 63.1 nM T20891 CC6PZ4 51354328 IC50 = 50.12 nM T20891 C2FVX4 51354329 IC50 = 630.96 nM T20891 CV06QD 51354330 IC50 = 1000 nM T20891 CR3AC1 51354331 IC50 = 25.12 nM T20891 CUXD62 51354613 IC50 = 0.631 nM T20891 C3G1VK 51354899 IC50 = 1258.93 nM T20891 CK7NP1 51354900 IC50 = 1000 nM T20891 CEDN75 51354901 IC50 = 1258.93 nM T20891 CB0EU1 51355190 IC50 = 125.89 nM T20891 C6K2SX 51356289 IC50 = 1000 nM T20891 C31WVJ 51356290 IC50 = 19952.62 nM T20891 CQ8T2R 51356291 IC50 = 7943.28 nM T20891 C9O7SG 51356292 IC50 = 12589.25 nM T20891 CYZ03E 51356852 IC50 = 251.19 nM T20891 CL3S8F 51356853 IC50 = 79.43 nM T20891 C67DUF 51356854 IC50 = 125.89 nM T20891 CAU2F6 51356855 IC50 = 501.19 nM T20891 CD07RV 51356856 IC50 = 251.19 nM T20891 CFM5I7 51357137 IC50 = 199.53 nM T20891 CP6R5J 51357138 IC50 = 125.89 nM T20891 CWCJ29 51357417 IC50 = 31.62 nM T20891 CS9WE1 51357418 IC50 = 63.1 nM T20891 C5G7BY 51357419 IC50 = 125.89 nM T20891 CBM4P9 51357696 IC50 = 794.33 nM T20891 C65MXB 51357954 IC50 = 7.943 nM T20891 C9IG1K 53317177 IC50 = 145000 nM T20891 C6VZ2R 53317178 IC50 = 13600 nM T20891 C6DNL1 53319793 IC50 = 7280 nM T20891 CI7RW5 53322416 IC50 > 25100 nM T20891 C9RIY1 53488414 Ki = 35 nM T20891 CRN28X 54581311 IC50 = 0.7943 nM T20891 C4Z0OC 56834890 Ki = 0.7 nM T20891 C67TJQ 56834891 Ki = 1.4 nM T20891 CFU89P 56926597 Ki = 2 nM T20891 C32CID 56926598 Ki = 0.6 nM T20891 CVO3R6 56926599 Ki = 0.9 nM T20891 CV8Z5C 56926697 Ki = 1.3 nM T20891 CO43FQ 56926699 Ki = 2.5 nM T20891 C4GT2U 56926701 Ki = 1 nM T20891 CAK91L 56955954 IC50 > 3600 nM T20891 C16RBI 57393424 IC50 = 390 nM T20891 CE4FA1 57396924 IC50 = 98 nM T20891 CLI7S3 57403897 IC50 = 150 nM T20891 CT70FI 59225251 IC50 = 68 nM T20891 CXJ63M 59603829 IC50 = 53 nM T20891 CQEU96 59603842 IC50 = 20 nM T20891 COH62U 60097413 IC50 > 10000 nM T20891 C1MR8Q 60097495 IC50 > 10000 nM T20891 CSZA16 60155724 IC50 > 3600 nM T20891 C9M4SZ 66759095 EC50 = 13000 nM T20891 C3YJ9P 66759299 EC50 = 30200 nM T20891 C7MJ5W 66760004 EC50 = 85800 nM T20891 C1HSE0 67035086 IC50 = 8200 nM T20891 CWI6K5 67035106 IC50 > 10000 nM T20891 C38RGB 67035556 IC50 = 9400 nM T20891 C8HOZ9 67041250 IC50 = 84 nM T20891 CV63UL 67240318 IC50 > 10000 nM T20891 C8I7GC 68293638 IC50 > 10000 nM T20891 CD56XK 68293660 IC50 = 6800 nM T20891 CDB62K 70681398 IC50 = 260 nM T20891 CN6GK4 70681405 IC50 = 75 nM T20891 C7GU5Q 70681406 IC50 = 220 nM T20891 C0NFK3 70683494 IC50 = 970 nM T20891 CG3C0B 70683495 IC50 = 400 nM T20891 CDFX37 70683509 IC50 = 84 nM T20891 C0WE8F 70685596 IC50 = 280 nM T20891 CKW18V 70685615 IC50 = 79 nM T20891 C9EV3Y 70685616 IC50 = 3300 nM T20891 C0E9RU 70687747 IC50 = 1200 nM T20891 CYHA21 70687748 IC50 = 110 nM T20891 CVPZ27 70687761 IC50 = 4500 nM T20891 C4BSI9 70689798 IC50 = 410 nM T20891 CTI38V 70691938 IC50 = 170 nM T20891 CU07RJ 70691948 IC50 = 46 nM T20891 CKT60L 71455860 Ki = 71 nM T20891 C8OWL6 71456015 IC50 = 220 nM T20891 CYN6R5 71461446 IC50 = 130 nM T20891 C2FAE3 71716356 IC50 = 26.5 nM T20891 CKN8U2 71718794 IC50 = 5700 nM T20891 C4B5RW 72725141 IC50 = 980 nM T20891 C1HW4B 89735655 IC50 = 330 nM T20891 CX6RP7 90160216 IC50 > 10000 nM T20891 C1ZY9N 102140491 IC50 = 1200 nM T20891 C3N8FE 102140492 IC50 = 4900 nM T20891 CY7BI2 118706214 IC50 > 10000 nM T20891 CV1KR7 119081690 IC50 = 17000 nM T20891 CMW6H9 121272820 IC50 = 6810 nM T20891 CYM25X 121276974 IC50 = 310 nM T20891 C0FKN9 124126383 IC50 = 6680 nM T20891 CP6KX0 124126392 IC50 = 512 nM T20891 CH8C5F 124126397 IC50 = 416 nM T20891 CCI5B4 124126403 IC50 = 112 nM T20891 C4MU2C 124126413 IC50 = 1520 nM T20891 C9E5FJ 127048247 IC50 = 26.5 nM T20891 CO1P3R 127049686 IC50 > 10000 nM T20891 C9CW6B 127049687 IC50 > 10000 nM T20891 C2AN7T 134611886 IC50 > 100000 nM T20891 C9FUK2 135151360 IC50 > 8300 nM T20891 C6RJD5 135400705 IC50 = 55000 nM T20891 CTR37Z 135408753 IC50 = 345000 nM T20891 CUN24C 135413416 IC50 = 15000 nM T20891 CXMS63 135417422 IC50 = 492000 nM T20891 C0O6UZ 135421655 IC50 = 86000 nM T20891 CG7V9T 135439636 IC50 = 461000 nM T20891 C2NX6D 135463111 IC50 = 122000 nM T20891 C9CWK6 135515802 IC50 = 472000 nM T20891 CO9SP6 135566717 IC50 = 6700 nM T20891 CSV20M 135567140 IC50 = 93000 nM T20891 CF74GJ 135820145 IC50 = 10900 nM T20891 C1PCJ3 136042251 IC50 = 1600 nM T20891 CG4KZ6 136060648 IC50 = 200 nM T20891 CSU8B2 136118610 EC50 = 76.7 nM T20891 CFK3J2 136228210 IC50 = 5200 nM T20891 C8OE2A 136232539 IC50 = 200 nM T20891 C93DEZ 136232540 IC50 = 200 nM T20891 C73ONP 136232541 IC50 = 800 nM T20891 CX8AS7 136232542 IC50 = 400 nM T20891 CBP49U 136232543 IC50 = 1200 nM T20891 CQ73OX 136232544 IC50 = 300 nM T20891 CY9C7I 136232545 IC50 = 1200 nM T20891 C5AE2Q 136232546 IC50 = 400 nM T20891 C7K8GH 136232547 IC50 = 900 nM T20891 CR98UF 136232548 IC50 = 8800 nM T20891 CO2J7M 136232549 IC50 = 15300 nM T20891 C03EOL 136232550 IC50 = 30300 nM T20891 C7LR6O 136232553 IC50 = 12400 nM T20891 CD51AZ 136232554 IC50 = 53900 nM T20891 C5MXA7 136232557 EC50 = 75.6 nM T20891 CC94GA 136244204 IC50 = 95000 nM T20891 CTD60C 136254211 IC50 = 33000 nM T20891 CSV87W 136254212 IC50 = 154000 nM T20891 CBK57T 136254213 IC50 = 109000 nM T20891 C9Q2VL 136254214 IC50 = 11000 nM T20891 CKW2Q9 136254215 IC50 = 39000 nM T20891 CJYB89 136254216 IC50 = 106000 nM T20891 CG42CK 136272415 IC50 = 5200 nM T20891 C6VB3O 145925651 IC50 >= 5000 nM T20891 C2MD1Q 155513187 IC50 > 10000 nM T20891 C86HPW 155518524 IC50 = 11000 nM T20891 D00ATA 5908088 IC50 = 520 nM T20891 D06BFH 1820 IC50 = 297000 nM T20891 D08KSQ 11637090 IC50 = 5900 nM T20891 D09EAE 10131254 IC50 = 1100 nM T20891 D0CM6T 11314340 Ki > 20000 nM T20891 D0EU1R 46215815 IC50 = 2.512 nM T20891 D0F5EI 10017019 IC50 = 12000 nM T20891 D0Q3KS 9957049 IC50 > 10000 nM T20891 D0S3TJ 76098 IC50 = 92000 nM T20891 D0V6GX 11311693 IC50 = 18 nM T41750 CZN6S9 743974 IC50 > 50118.72 nM T41750 CS02XG 9871912 IC50 = 389 nM T41750 CF6AV4 9914410 IC50 = 1392 nM T41750 CP96LK 9916972 IC50 = 145 nM T41750 CHSN85 9985258 IC50 = 990 nM T41750 CGEJ24 9985625 IC50 = 7500 nM T41750 CF86IP 10030697 IC50 = 410 nM T41750 C6L7UO 10032265 IC50 = 359 nM T41750 COC68H 10053841 IC50 = 3000 nM T41750 CXFW65 10053886 IC50 = 460 nM T41750 CR6NW9 10054055 IC50 = 430 nM T41750 C4P6KU 10077369 IC50 = 6000 nM T41750 CK05GO 10097880 IC50 = 910 nM T41750 C0P5DE 10144347 IC50 = 411 nM T41750 C0B5WP 10144633 IC50 = 74 nM T41750 C62RYU 10144925 IC50 = 445 nM T41750 CFD96W 10145290 IC50 = 3020 nM T41750 C70HKJ 10145603 IC50 = 279 nM T41750 CTR46Q 10167904 IC50 = 12 nM T41750 C85IFN 10168348 IC50 = 83 nM T41750 C6CH8L 10210150 IC50 = 315 nM T41750 CQ0NT1 10211765 IC50 = 380 nM T41750 C4S9MD 10211943 IC50 = 497 nM T41750 C0B2DH 10231964 IC50 = 701 nM T41750 C8CNK1 10232009 IC50 = 93 nM T41750 C8R7YJ 10255803 IC50 > 20000 nM T41750 C08BCM 10257357 IC50 = 64 nM T41750 CDZ62K 10257629 IC50 = 390 nM T41750 CQ49SX 10280734 IC50 = 406 nM T41750 CMW97S 10282059 IC50 = 216 nM T41750 CW16YI 10282162 IC50 = 277 nM T41750 C09YQC 10282370 IC50 = 198 nM T41750 CMK7Q6 10324097 IC50 = 2100 nM T41750 CI4G2Z 10369244 IC50 > 25000 nM T41750 CO5PW3 10369510 IC50 = 220 nM T41750 C1V8EH 10393937 IC50 = 480 nM T41750 CRCP21 10415723 IC50 = 7100 nM T41750 C0BJQ4 10436553 IC50 = 2800 nM T41750 CC1FQ2 10461010 IC50 > 10000 nM T41750 CF8I6B 10483282 IC50 = 98 nM T41750 CO2CQ7 11331120 IC50 = 370 nM T41750 CC5WD2 11444850 IC50 = 290 nM T41750 CJ4K2U 11456187 IC50 = 510 nM T41750 C0N6UB 11527207 IC50 = 795 nM T41750 CB59HM 11570626 IC50 = 1019 nM T41750 CR78YS 11585375 IC50 = 378 nM T41750 C3JE1T 11585452 IC50 = 1134 nM T41750 C1BT6K 11592461 IC50 = 885 nM T41750 CCQZ38 11621378 IC50 = 933 nM T41750 CW8LD3 11657413 IC50 = 711 nM T41750 CLY98H 11678967 IC50 = 1984 nM T41750 C4B2JQ 11699553 IC50 = 4337 nM T41750 C3RZF0 11756248 IC50 = 7400 nM T41750 CU56HZ 11757679 IC50 = 5700 nM T41750 CE0CZ6 11764614 IC50 = 373 nM T41750 CSZQ52 11764615 IC50 = 87 nM T41750 CK25CM 11949739 IC50 = 2023 nM T41750 CTM6N5 11949740 IC50 = 4256 nM T41750 CNI85P 11950075 IC50 = 286 nM T41750 CL2GD7 11950794 IC50 = 178 nM T41750 CSV4A0 11950795 IC50 = 171 nM T41750 C6BYQ0 11950971 IC50 = 217 nM T41750 CM2XR7 11950972 IC50 = 117 nM T41750 C7H2SG 11952035 IC50 = 296 nM T41750 CQ0KU7 11952211 IC50 = 132 nM T41750 C1SJ5W 11952213 IC50 = 610 nM T41750 C3A7CL 11952214 IC50 = 118 nM T41750 C7VI6D 11952394 IC50 = 3525 nM T41750 COF34S 16100296 IC50 = 28.3 nM T41750 C05PIH 16100300 IC50 = 93 nM T41750 C53GHR 16100334 IC50 = 38 nM T41750 CGC2I1 20775791 IC50 > 1000 nM T41750 CB7ID8 20775792 IC50 > 1000 nM T41750 C29FRA 20775916 IC50 = 638 nM T41750 C97VQA 20776096 IC50 = 732 nM T41750 CSH17F 20776097 IC50 = 645 nM T41750 CK91GP 22496358 IC50 = 429 nM T41750 CQ42EI 22496365 IC50 = 207 nM T41750 CMVS81 22496371 IC50 = 368 nM T41750 C4KL3V 22496373 IC50 = 1113 nM T41750 CKXG15 22496384 IC50 = 381 nM T41750 C1YAO5 22496395 IC50 = 729 nM T41750 CG45BT 22496412 IC50 = 721 nM T41750 C86YBZ 22496431 IC50 = 1002 nM T41750 CPRG93 22496441 IC50 > 1000 nM T41750 CZR6D0 22496445 IC50 = 770 nM T41750 CFE72V 22496448 IC50 = 316 nM T41750 C7NZ5H 22496449 IC50 = 290 nM T41750 CRI13U 22496451 IC50 = 777 nM T41750 CCI62H 22496457 IC50 = 320 nM T41750 C49VUW 22496459 IC50 = 510 nM T41750 CK78ZG 22496477 IC50 = 390 nM T41750 CSV48P 22496546 IC50 = 584 nM T41750 CE8UB0 22496557 IC50 = 293 nM T41750 C7JW4V 23550062 IC50 = 45 nM T41750 C03JNO 42617999 IC50 = 565 nM T41750 C8HOD7 44431020 IC50 = 1279 nM T41750 CQS1U6 45485585 EC50 > 10000 nM T41750 CFTG29 53323247 IC50 = 4100 nM T41750 CFU20M 53325823 IC50 > 10000 nM T41750 CG2M3A 53325824 IC50 > 25000 nM T41750 CD2X1W 53469443 IC50 = 2100 nM T41750 C6TEK8 54765284 IC50 = 1500 nM T41750 C0T3KY 54765285 IC50 = 1400 nM T41750 CH8P3M 57391489 IC50 = 1600 nM T41750 CZ07MU 57391686 Ki = 300 nM T41750 CW4FM5 57393425 Ki = 1950 nM T41750 C7T0OK 57393426 Ki = 152 nM T41750 CIU91X 57396928 Ki = 939 nM T41750 C4AJ1G 57403703 IC50 = 1100 nM T41750 C4WM0U 57518490 IC50 = 307 nM T41750 CYUG59 60170767 IC50 = 3370 nM T41750 C6IV0K 60170855 IC50 = 478 nM T41750 CSN5C8 60170856 IC50 = 753 nM T41750 C4MKG9 60170857 IC50 = 431 nM T41750 CPLU74 60170970 IC50 = 1844 nM T41750 CX19CT 60170971 IC50 = 2419 nM T41750 CA0EO3 60171059 IC50 = 1336 nM T41750 C5JLE4 60171060 IC50 = 4996 nM T41750 CQ6O3H 60171061 IC50 = 2056 nM T41750 C2H1OF 60171062 IC50 = 1684 nM T41750 CB53RK 122189577 IC50 = 1400 nM T41750 CDAO27 122189708 IC50 = 1100 nM T41750 CEQ09Z 122189709 IC50 = 1000 nM T41750 CS1D9R 122189714 IC50 = 750 nM T41750 CL0AR4 122189722 IC50 = 1300 nM T41750 C7N3KL 145960401 EC50 = 0.0582 nM T41750 C92BLJ 145960433 EC50 = 0.0397 nM T41750 C0X5MI 145960850 EC50 = 2.032 nM T41750 C1ZNU5 145961751 EC50 = 0.189 nM T41750 CW90YV 145962263 EC50 = 177 nM T41750 CN9CR1 145962270 EC50 = 0.224 nM T41750 CA29XQ 145962515 EC50 = 1.16 nM T41750 CVQ62L 145962554 EC50 = 2.032 nM T41750 C97HKT 145962593 EC50 = 1.21 nM T41750 CGO8V1 145962872 EC50 = 0.102 nM T41750 C0ADY2 145962907 EC50 = 114 nM T41750 CLO0S4 145967618 EC50 = 0.867 nM T41750 C3JW1P 145968295 EC50 = 2.691 nM T41750 C0T1ZE 145968501 EC50 = 2.032 nM T41750 C0ZTW8 145968513 EC50 = 1.103 nM T41750 CMB10N 145969232 EC50 = 1.654 nM T41750 C5J8HP 145969289 EC50 = 6.26 nM T41750 C7UZT9 145969722 EC50 = 2.194 nM T41750 CS36QG 145969945 EC50 = 6.258 nM T41750 C3AI9B 145970440 EC50 = 5.53 nM T41750 CX0C6A 145970613 EC50 = 1.646 nM T41750 CCZ9K7 145970869 EC50 = 0.133 nM T41750 CDB15L 145971098 EC50 = 5.828 nM T41750 CN4Z2C 145971132 EC50 = 0.812 nM T41750 CC3Y2Z 145987495 EC50 = 3.545 nM T74937 C4WNY9 21632 IC50 = 50000 nM T74937 C0Z3RY 36917 IC50 = 2000 nM T74937 CGM60S 128646 IC50 = 3000 nM T74937 C9ZEB3 667838 IC50 = 33113.11 nM T74937 C9B4GC 3035523 IC50 = 2570.4 nM T74937 CTX1E7 10059965 IC50 = 52480.75 nM T74937 C1V9HD 10263758 IC50 = 74.13 nM T74937 CB2S7I 10398787 IC50 = 1202.26 nM T74937 CA1TR3 10443390 IC50 = 1000000 nM T74937 C9H0WQ 13477989 IC50 = 204173.79 nM T74937 C93PIT 13477996 IC50 = 83176.38 nM T74937 C8DYA7 14450863 IC50 = 36307.81 nM T74937 CEMA54 14576743 IC50 = 46773.51 nM T74937 CT4EX2 14576744 IC50 = 199526.23 nM T74937 CJ14BA 15124054 IC50 = 74131.02 nM T74937 C3QH8N 15124056 IC50 = 30902.95 nM T74937 CS3L6P 15124057 IC50 = 120226.44 nM T74937 C5WQF1 15124058 IC50 = 2398.83 nM T74937 CP9K6X 15124059 IC50 = 707945.78 nM T74937 C76YKQ 15124060 IC50 = 354813.39 nM T74937 CL7VQ4 15124061 IC50 = 97723.72 nM T74937 CKZ8B2 15124062 IC50 = 95499.26 nM T74937 C7GY6A 15124063 IC50 = 52480.75 nM T74937 CBO90P 15124064 IC50 = 28183.83 nM T74937 CZ5F4U 15124065 IC50 = 16982.44 nM T74937 CIK3Y6 15124066 IC50 = 12022.64 nM T74937 C5EW7A 15124067 IC50 = 5623.41 nM T74937 CUEG95 15124068 IC50 = 46773.51 nM T74937 C09FCN 15124070 IC50 = 75857.76 nM T74937 CN5P4L 15124071 IC50 = 102329.3 nM T74937 C6HEF5 18990372 IC50 = 50000 nM T74937 CRGB58 18990395 IC50 = 50000 nM T74937 CYD3Q1 20070445 IC50 = 354813.39 nM T74937 CJ2B1A 20070452 IC50 = 173780.08 nM T74937 C3SK4Z 20070458 IC50 = 154881.66 nM T74937 CD7KH6 23274107 IC50 = 1513.56 nM T74937 C8Y7MP 25880073 IC50 = 147910.84 nM T74937 CJ8O6A 25880076 IC50 = 74131.02 nM T74937 CPG7N4 43555101 IC50 = 338844.16 nM T74937 C3NF5L 44306283 IC50 = 338844.16 nM T74937 CW8V9R 44306284 IC50 = 501187.23 nM T74937 CJ3ZM4 44306413 IC50 = 147910.84 nM T74937 CU8O9E 44306481 IC50 = 12022.64 nM T74937 CJ2T6Q 44306637 IC50 = 48977.88 nM T74937 CX8J1U 44306773 IC50 = 61659.5 nM T74937 C8D9ES 44306876 IC50 = 676.08 nM T74937 C1A9FU 44306901 IC50 = 158489.32 nM T74937 C5HY1D 44306902 IC50 = 1995.26 nM T74937 CP15DR 44306916 IC50 = 2187.76 nM T74937 C61ERI 44307011 IC50 = 575439.94 nM T74937 CS6G7L 44307012 IC50 = 69183.1 nM T74937 CVNY04 44307075 IC50 = 114815.36 nM T74937 D0D7GL 10789 IC50 = 2000 nM T85435 D03ZBT 11626560 IC50 = 102 nM T85435 D04LVK 57379345 IC50 = 7 nM T85435 D07POC 176870 IC50 > 12500 nM T85435 D08CDI 208908 IC50 = 17000 nM T85435 D08PIE 68165256 IC50 = 196 nM T85435 D09XZB 123631 IC50 > 50000 nM T85435 D0B0AX 5328127 IC50 > 50000 nM T85435 D0E6XR 3062316 IC50 > 50000 nM T85435 D0EG1I 9926791 IC50 > 10000 nM T85435 D0O8GK 71496458 IC50 = 912 nM T85435 D0R0MW 5329102 IC50 = 3200 nM T85435 D0W5HK 216239 IC50 = 5300 nM T85435 D01GFX 11640390 IC50 = 16 nM T85435 D01HKZ 57345941 IC50 = 231 nM T85435 D02QWY 24785538 IC50 = 1.7 nM T85435 D02RJY 11442891 IC50 > 10000 nM T85435 D03HUX 49792852 IC50 > 10000 nM T85435 D03LWG 53235510 IC50 = 3371 nM T85435 D07DTV 11338033 IC50 > 10000 nM T85435 D07EHV 44814409 IC50 > 10000 nM T85435 D07HPJ 11476171 IC50 = 244 nM T85435 D0E3TC 44259 IC50 = 8.5 nM T85435 D0N6NM 71721648 IC50 = 65 nM T85435 D0O0LS 25141092 IC50 = 209 nM T85435 D0O6WV 24794418 IC50 > 2000 nM T85435 D0O9PQ 57390074 IC50 = 100 nM T85435 D0P1CV 46191454 IC50 > 10000 nM T85435 D0Q9UX 16718576 IC50 > 10000 nM T85435 D0VF6E 1401 IC50 > 50000 nM T85435 D0WS1V 448991 IC50 = 2200 nM T85435 D00PWQ 3820 IC50 > 100000 nM T85435 D0YK9D 9956119 IC50 > 10000 nM T85435 D09HEV 6539952 IC50 > 20000 nM T85435 D0H4GI 10275001 IC50 > 10000 nM T85435 D0IT6Q 3038522 IC50 > 30000 nM T85435 D0T3ME 156422 IC50 > 30000 nM T85435 CH21PG 2428 IC50 > 50000 nM T85435 CN1HZ8 77390 IC50 = 700 nM T85435 C63WLY 89644 IC50 > 10 ug.mL-1 T85435 C5JE2Z 104860 IC50 = 9.4 ug.mL-1 T85435 CI82CW 147317 IC50 = 10 nM T85435 CRFU83 156413 IC50 > 50000 nM T85435 CI1NA5 159926 IC50 = 3.5 ug.mL-1 T85435 CYBA43 177458 IC50 = 3.9 ug.mL-1 T85435 C1ZG2U 449087 IC50 > 10000 nM T85435 CL42EI 577406 IC50 = 1300 nM T85435 C2VRY5 1204889 IC50 > 100000 nM T85435 CXBF05 1204893 IC50 > 100000 nM T85435 CFN1X5 1205024 IC50 > 100000 nM T85435 C07AHW 1205040 IC50 > 100000 nM T85435 CKNO43 1205381 IC50 = 28000 nM T85435 C9H7DW 1205672 IC50 = 19500 nM T85435 C5PDS4 1206018 IC50 > 100000 nM T85435 CYG3F7 1206240 IC50 > 100000 nM T85435 C8TM4R 1206252 IC50 > 100000 nM T85435 C59JUN 1206254 IC50 = 57600 nM T85435 CAM8U9 1206256 IC50 = 27300 nM T85435 CSN92F 1206261 IC50 > 100000 nM T85435 CLAH32 1206264 IC50 > 100000 nM T85435 C0H3WZ 1206279 IC50 > 100000 nM T85435 CPV94W 1218955 IC50 = 905 nM T85435 C6IZE0 1225146 IC50 > 100000 nM T85435 CY17ZI 1227452 IC50 > 100000 nM T85435 C9ZW7G 1230091 IC50 > 100000 nM T85435 C90KON 1231530 IC50 > 100000 nM T85435 C1I2UP 1232262 IC50 > 100000 nM T85435 C5TSE1 1232814 IC50 > 100000 nM T85435 C9Y0JC 1237187 IC50 > 100000 nM T85435 CON65H 1565908 IC50 > 100000 nM T85435 CBV04C 1731052 IC50 = 79500 nM T85435 CG1FL5 1731078 IC50 > 100000 nM T85435 CPVD46 1774817 IC50 > 100000 nM T85435 CCN9D5 3142817 IC50 = 900 nM T85435 CPT61U 5328112 IC50 > 50000 nM T85435 CXR9K1 5328115 IC50 > 50000 nM T85435 CM0H5O 5328117 IC50 > 50000 nM T85435 CDM98R 5328125 IC50 > 50000 nM T85435 CDY2O3 5328134 IC50 > 50000 nM T85435 CC1O0M 5328135 IC50 > 50000 nM T85435 C14LVT 5328137 IC50 > 50000 nM T85435 COT45A 5328149 IC50 > 50000 nM T85435 CDV19S 5328354 IC50 > 50000 nM T85435 C1D0YT 5328357 IC50 > 50000 nM T85435 CC4O6Y 5328360 IC50 > 50000 nM T85435 CFW19M 5329009 IC50 = 2600 nM T85435 CSY10K 5329111 IC50 > 50000 nM T85435 CZ3LK2 5330387 IC50 = 1690 nM T85435 CRU94N 5330388 IC50 > 10000 nM T85435 CDB68F 5330389 IC50 > 10000 nM T85435 C7CX0H 5330390 IC50 = 10000 nM T85435 C8E0XS 5330391 IC50 > 10000 nM T85435 CW1VX9 5330392 IC50 > 10000 nM T85435 CF01JS 5330804 IC50 = 2400 nM T85435 CDQ3M7 5359485 IC50 = 2.1 ug.mL-1 T85435 C54BYP 5360741 IC50 = 7.9 ug.mL-1 T85435 CM7Z4V 5378081 IC50 = 1200 nM T85435 CZ2NG9 5473542 IC50 = 3 nM T85435 C7GD1T 5753500 IC50 = 36300 nM T85435 CB7WK3 5938113 IC50 > 100000 nM T85435 CEOT94 6155669 IC50 = 65300 nM T85435 C5NAI6 6183972 IC50 = 6 nM T85435 C2OL7K 9796455 IC50 = 33000 nM T85435 CM5Z8X 9869943 IC50 > 100000 nM T85435 C0YM9T 9870827 IC50 = 83 nM T85435 CPQ13K 9933545 IC50 = 24000000 nM T85435 CN0AJ9 9934347 IC50 = 40 nM T85435 C2W3AV 9995236 IC50 = 80000 nM T85435 CUJR40 10062694 EC50 > 2000 nM T85435 CC78NE 10179293 IC50 = 3 nM T85435 CSGD16 10246246 IC50 > 7000 nM T85435 CC9E5Q 10249989 IC50 = 420 nM T85435 CJGH26 10275985 IC50 = 24 nM T85435 C7SFI1 10296883 IC50 > 10000 nM T85435 C7HBP6 10429593 IC50 > 10000 nM T85435 COB2X8 10602350 IC50 > 50000 nM T85435 CJO8Q1 10738332 IC50 > 50000 nM T85435 CRK56F 11237786 IC50 > 6000 nM T85435 CBOP58 11293798 Ki > 10000 nM T85435 CJ8A6Y 11341428 IC50 > 6000 nM T85435 C26BZX 11362471 Ki > 10000 nM T85435 CWXB93 11397177 Ki > 10000 nM T85435 CEP8N2 11489351 IC50 > 6000 nM T85435 CU13WV 11518389 IC50 > 50000 nM T85435 CL7X4Q 11530963 IC50 = 23000 nM T85435 CQ06DZ 11532796 IC50 = 27300 nM T85435 CTG83F 11539329 Ki > 5200 nM T85435 CWHK97 11553173 IC50 > 40000 nM T85435 CACS26 11561968 Ki > 2000 nM T85435 CKO0G8 11568821 IC50 > 40000 nM T85435 CMN1Q3 11569457 IC50 = 33500 nM T85435 CDT68P 11576099 IC50 = 7000 nM T85435 CQOI76 11576375 IC50 = 9500 nM T85435 CO9KP5 11583459 IC50 = 76 nM T85435 C5DHZ2 11590126 IC50 = 13800 nM T85435 CMIL86 11590363 Ki > 5200 nM T85435 C43JZU 11604436 IC50 = 4800 nM T85435 CGU7N0 11604739 Ki = 5300 nM T85435 CYA04X 11605000 IC50 > 40000 nM T85435 C9T6SC 11640926 Ki > 5200 nM T85435 CU38TK 11649146 IC50 = 68 nM T85435 CJ97KW 11655878 IC50 > 40000 nM T85435 CAJS96 11662893 Ki = 9000 nM T85435 CKAH36 11669784 IC50 = 3600 nM T85435 CU0E8O 11690457 Ki > 2000 nM T85435 C6EOL3 11691146 IC50 = 32500 nM T85435 CTRZ62 11705264 IC50 > 40000 nM T85435 CA2KE3 11719817 IC50 = 16000 nM T85435 C45EWD 11723489 IC50 > 7000 nM T85435 CP7AH3 11755812 IC50 = 50000 nM T85435 C9JT4S 11847343 IC50 = 7012 nM T85435 CXK1C3 12755122 IC50 = 1200 nM T85435 C5KN4X 13973144 IC50 = 60 nM T85435 CDGF78 15282555 IC50 = 2900 nM T85435 C0M7TW 15948947 IC50 = 7631 nM T85435 C1VNB4 15948949 IC50 = 746 nM T85435 CH8ZG5 15949048 IC50 = 588 nM T85435 CK2Z6Y 15949521 IC50 = 1493 nM T85435 CBZF29 15949522 IC50 = 1988 nM T85435 C34MCY 15949523 IC50 = 409 nM T85435 CS3P9G 15949524 IC50 = 63 nM T85435 C1KPH2 15949525 IC50 = 3332 nM T85435 C7LB4I 15949613 IC50 > 10000 nM T85435 C5JG9R 15949617 IC50 = 4 nM T85435 C8FT6U 15949618 IC50 = 1961 nM T85435 C30PVQ 15949619 IC50 = 75 nM T85435 C3PNO2 15949620 IC50 = 818 nM T85435 C4I5RS 15949621 IC50 > 10000 nM T85435 CVJ9A0 15949712 IC50 = 2345 nM T85435 CEI2K8 15949887 IC50 = 5165 nM T85435 CAIN63 15949888 IC50 > 10000 nM T85435 C2VDI1 15949889 IC50 = 4401 nM T85435 COC02T 15949890 IC50 = 1613 nM T85435 CFQ6X3 15949974 IC50 = 1435 nM T85435 CMKZ23 15949975 IC50 = 1141 nM T85435 CWM5L4 15949976 IC50 = 3162 nM T85435 CO7NG2 15950141 IC50 = 3012 nM T85435 COIG45 15950224 IC50 = 661 nM T85435 C9V0TO 15950311 IC50 > 10000 nM T85435 CFPW41 16007116 Ki > 5200 nM T85435 CQR5O7 16042971 IC50 > 10000 nM T85435 CH7MS6 16059729 IC50 > 42000 nM T85435 CQG45C 16109001 IC50 = 4200 nM T85435 C1U8XW 16109036 IC50 = 2900 nM T85435 C5VPH9 16129448 IC50 = 502 nM T85435 CVZK29 16223008 IC50 > 50000 nM T85435 CJ5KU9 16659012 IC50 = 610 nM T85435 C2IF3P 16678352 IC50 = 22600 nM T85435 C3IO1C 16679060 IC50 > 30000 nM T85435 C9IW5S 16730105 IC50 = 24000 nM T85435 CPRM54 18830136 IC50 = 8 nM T85435 CNQ18K 19596882 IC50 = 340 nM T85435 C8TYO5 19596902 IC50 = 130 nM T85435 C4S6OW 19596919 IC50 = 6000 nM T85435 CJMG54 19596932 IC50 = 80 nM T85435 CQOS58 19596969 IC50 > 100000 nM T85435 CP17NS 19596973 IC50 = 12 nM T85435 CH4B5K 21081523 IC50 > 5000 nM T85435 C25UKC 21081761 IC50 > 5000 nM T85435 C6JV7W 23400934 IC50 > 7000 nM T85435 CD5S7O 23401001 IC50 > 7000 nM T85435 CF67IQ 23628269 IC50 = 140 nM T85435 CQHK69 23646624 IC50 = 1000 nM T85435 C2RV3U 24180608 IC50 > 30000 nM T85435 CA3I4T 24753787 IC50 > 50000 nM T85435 C7YG1N 24759534 IC50 = 55000 nM T85435 CAJ4T2 24762205 IC50 > 10000 nM T85435 CQNP54 24764449 IC50 = 1000 nM T85435 CCPS81 24764502 IC50 > 35000 nM T85435 C81GVC 24774737 IC50 = 3162.28 nM T85435 CN8R5S 24779728 IC50 = 23 nM T85435 C9B2TF 24880043 IC50 = 3700 nM T85435 C4V9GH 24894117 IC50 = 43000 nM T85435 CJH19T 24894883 IC50 = 47000 nM T85435 CB5TP8 24894992 IC50 = 27000 nM T85435 CFW40U 24894997 IC50 = 44000 nM T85435 CN13JF 24899915 IC50 = 2.9 ug.mL-1 T85435 CBWR97 24899916 IC50 = 1.3 ug.mL-1 T85435 C9F2JD 24899917 IC50 > 10 ug.mL-1 T85435 C64MTI 24900160 IC50 = 3 ug.mL-1 T85435 CO2I6Q 24900161 IC50 = 8.1 ug.mL-1 T85435 C5FD1A 24937369 IC50 = 19800 nM T85435 C6MP4L 24986245 EC50 = 241 nM T85435 C4AQ3M 24986600 EC50 = 14 nM T85435 CA4W7M 24987312 EC50 = 582 nM T85435 CS7UK9 24987314 EC50 = 4170 nM T85435 CLA59H 24987650 EC50 = 126 nM T85435 C3O9SV 24987652 EC50 = 320 nM T85435 C4EG8R 24993189 IC50 > 10000 nM T85435 C2ICS7 25065806 IC50 > 1000 nM T85435 CSNC57 25110758 IC50 > 6000 nM T85435 C0GOX5 25110759 IC50 = 5600 nM T85435 CC2R7S 25110760 IC50 > 10000 nM T85435 CL82CU 25110796 IC50 = 3900 nM T85435 C4OA5D 25113170 IC50 = 1.6 nM T85435 CTV54O 25123227 IC50 > 10000 nM T85435 CG3XC9 25124150 Ki = 2.2 nM T85435 CO2IR5 25124816 Ki = 1.3 nM T85435 CP9LZ8 25157323 IC50 = 4 nM T85435 CS9G4P 25157326 IC50 = 34 nM T85435 C3VR6L 25157614 IC50 = 10 nM T85435 C10CVP 25160012 IC50 = 339 nM T85435 CUAB05 25160153 IC50 = 375.3 nM T85435 CCM97P 25160155 IC50 = 349 nM T85435 CHT0B4 25169252 IC50 = 330 nM T85435 CJL25F 25169253 IC50 = 1500 nM T85435 C8IX5P 25174241 IC50 = 462 nM T85435 CTKC48 25174394 IC50 = 9866 nM T85435 CE6PB7 25175712 IC50 = 1806 nM T85435 CB1Z8N 25175860 IC50 = 1303 nM T85435 CIHB16 25175861 IC50 = 427 nM T85435 CVO5B2 25175862 IC50 = 170 nM T85435 C04HDK 25176007 IC50 = 330 nM T85435 CT2K5R 25176014 IC50 = 41 nM T85435 C8A9EJ 25176163 IC50 = 3822 nM T85435 C6G7RT 25176165 IC50 = 189 nM T85435 CPM9Q8 25176330 IC50 = 3694 nM T85435 C81NBM 25176332 IC50 = 1764 nM T85435 CI58TS 25176649 IC50 = 1069 nM T85435 CSEN02 25176653 IC50 = 1190 nM T85435 C85KCS 25178328 IC50 = 5100 nM T85435 CIG4H0 25178539 IC50 = 2600 nM T85435 C4GI6J 25178540 IC50 = 6300 nM T85435 C2RX6E 25190503 IC50 = 560 nM T85435 CFN61D 25190504 IC50 > 6000 nM T85435 C8LQS3 25190505 IC50 > 6000 nM T85435 C20WQJ 25190506 IC50 > 6000 nM T85435 CM61RX 25190507 IC50 > 6000 nM T85435 C5UCN3 25190508 IC50 = 5800 nM T85435 CTVK31 25190509 IC50 > 6000 nM T85435 CY43QX 25190510 IC50 = 150 nM T85435 C09SGT 25190511 IC50 = 240 nM T85435 C9O0AL 25190512 IC50 = 6100 nM T85435 C6RC2N 25190513 IC50 = 1600 nM T85435 CA9U5F 25190514 IC50 > 6000 nM T85435 C1ZCK4 25190515 IC50 > 6000 nM T85435 CBX7Z3 25190516 IC50 > 6000 nM T85435 CY3X8L 25190517 IC50 > 6000 nM T85435 CONP02 25190518 IC50 = 380 nM T85435 CL81KR 25190519 IC50 = 630 nM T85435 C2I6JX 25190520 IC50 = 3800 nM T85435 C8TK1S 25190521 IC50 = 51 nM T85435 CHD51B 25190522 IC50 > 6000 nM T85435 C0G9EX 25190523 IC50 > 6000 nM T85435 CUJS83 25190524 IC50 > 6000 nM T85435 CE3W4R 25190525 IC50 > 6000 nM T85435 CIAB51 25190526 IC50 > 6000 nM T85435 CA4Z2Y 25190527 IC50 > 6000 nM T85435 C8OW9I 25190528 IC50 > 6000 nM T85435 C5PH6D 25190529 IC50 > 6000 nM T85435 CZ46JX 25190530 IC50 = 5200 nM T85435 CE3T5U 25190531 IC50 = 2400 nM T85435 CEHP95 25190532 IC50 > 6000 nM T85435 C06LXS 25190533 IC50 > 6000 nM T85435 C9RXL3 25190534 IC50 = 2000 nM T85435 CC1E3O 25190535 IC50 > 6000 nM T85435 C1NZ4D 25190536 IC50 > 6000 nM T85435 CNR75T 25190537 IC50 > 6000 nM T85435 C7LMI1 25190538 IC50 > 6000 nM T85435 CLU7D2 25190539 IC50 > 6000 nM T85435 CD2Z1T 25190540 IC50 > 6000 nM T85435 CUP7E4 25190541 IC50 > 6000 nM T85435 C57KGJ 25190542 IC50 > 6000 nM T85435 CF9C5J 25190543 IC50 > 6000 nM T85435 C3KJ6P 25190544 IC50 > 6000 nM T85435 CU6VA8 25190545 IC50 = 480 nM T85435 CR0JP6 25190546 IC50 = 3250 nM T85435 CJLB59 25190547 IC50 > 5000 nM T85435 C27RCT 25190548 IC50 = 970 nM T85435 CM7A8T 25190549 IC50 = 4000 nM T85435 C3YA7U 25190550 IC50 > 5000 nM T85435 C6SE7Y 25190551 IC50 > 5000 nM T85435 CPK7E0 25190552 IC50 > 5000 nM T85435 CA2K4Q 25190553 IC50 > 5000 nM T85435 CWRO62 25190554 IC50 > 5000 nM T85435 C5UFS2 25190555 IC50 > 5000 nM T85435 C6J2UZ 25190556 IC50 > 5000 nM T85435 CMP9A2 25190557 IC50 > 5000 nM T85435 CKP50F 25190558 IC50 = 1950 nM T85435 CE3W9P 25190559 IC50 = 4900 nM T85435 CNBO46 25190560 IC50 = 3300 nM T85435 CCP4K9 25190561 IC50 = 4300 nM T85435 CYK5Z2 25190562 IC50 = 2200 nM T85435 C25JMO 25190563 IC50 > 5000 nM T85435 CJ4W6E 25190564 IC50 > 5000 nM T85435 CBV3D6 25190565 IC50 = 3800 nM T85435 CE9UI6 25190566 IC50 > 5000 nM T85435 CAK4E6 25190567 IC50 = 4500 nM T85435 CTR6A2 25190568 IC50 = 3600 nM T85435 CC40BJ 25190569 IC50 > 5000 nM T85435 C7B6OS 25190570 IC50 > 5000 nM T85435 CCJY98 25190571 IC50 > 5000 nM T85435 C6FGQ1 25206346 IC50 > 10000 nM T85435 CNG96H 25210579 IC50 > 10000 nM T85435 CM0T8S 25210970 IC50 = 0.4 nM T85435 CO0RF6 25218593 IC50 = 6.3 nM T85435 C2TXC6 25218656 IC50 = 9300 nM T85435 CHO43Y 28491869 IC50 = 2080 nM T85435 CWDU21 39935257 IC50 = 27 nM T85435 CU53WB 42596953 IC50 = 3600 nM T85435 CJ5U1X 42639664 IC50 = 3.7 ug.mL-1 T85435 CTN41Y 44156909 IC50 > 10000 nM T85435 CN0X1C 44156917 IC50 > 10000 nM T85435 CC1P5L 44156965 IC50 = 1000 nM T85435 CB8YN2 44201333 IC50 = 160 nM T85435 CF9UB1 44219665 IC50 > 40000 nM T85435 CXPN30 44219666 IC50 > 40000 nM T85435 CVEU45 44219667 IC50 = 11100 nM T85435 CEL61X 44229839 IC50 > 10000 nM T85435 CW3BP8 44398371 IC50 = 9800 nM T85435 C4YMI9 44447890 IC50 > 1000 nM T85435 CR65PM 44447895 IC50 > 1000 nM T85435 C4B7KF 44515722 IC50 = 28.1 nM T85435 C8H4FA 44515723 IC50 = 726 nM T85435 CC7E4K 44564705 IC50 > 10000 nM T85435 C42ZEW 44564706 IC50 > 10000 nM T85435 C53MCK 44564747 IC50 > 10000 nM T85435 CDI31F 44564748 IC50 = 9700 nM T85435 CA17NT 44564749 IC50 > 10000 nM T85435 CMIZ20 44564750 IC50 > 10000 nM T85435 CSO9F8 44564751 IC50 > 10000 nM T85435 C8ATG9 44564787 IC50 > 10000 nM T85435 CM50GS 44564788 IC50 > 10000 nM T85435 C3Q0DX 44564789 IC50 = 6950 nM T85435 CP40XB 44564790 IC50 > 10000 nM T85435 C35NTB 44564791 IC50 > 10000 nM T85435 CJY83G 44564817 IC50 > 10000 nM T85435 CLK98G 44564818 IC50 > 10000 nM T85435 CF2D1K 44564819 IC50 > 10000 nM T85435 C3CQ9K 44564820 IC50 > 10000 nM T85435 CI8V2L 44564821 IC50 > 10000 nM T85435 C9PO7J 44564860 IC50 > 10000 nM T85435 C16FJW 44564861 IC50 > 10000 nM T85435 C8AMX5 44564862 IC50 = 2700 nM T85435 CTR59U 44564863 IC50 > 10000 nM T85435 C9EY4C 44564864 IC50 > 10000 nM T85435 CG5Z7T 44564910 IC50 > 10000 nM T85435 CU9O4C 44564911 IC50 > 10000 nM T85435 CXZ15S 44564954 IC50 = 630 nM T85435 CZ78WJ 44564955 IC50 = 2150 nM T85435 CJ1X9V 44565013 IC50 = 1600 nM T85435 CN2Q3D 44565014 IC50 = 940 nM T85435 CM2GN3 44565015 IC50 > 10000 nM T85435 C6RV9I 44565016 IC50 > 10000 nM T85435 CJC85A 44565069 IC50 = 7900 nM T85435 CWFB42 44571820 IC50 = 7 nM T85435 CJAV21 44573146 IC50 = 940 nM T85435 CP9E4J 44573266 IC50 > 5000 nM T85435 CLA24D 44573267 IC50 > 5000 nM T85435 C51CDF 44573268 IC50 = 350 nM T85435 CDT4K9 44573269 IC50 = 700 nM T85435 CD8Q5P 44573306 IC50 = 5500 nM T85435 C5CA0V 44573307 IC50 = 1700 nM T85435 CNMO98 44573308 IC50 = 480 nM T85435 CAZ59C 44573309 IC50 = 400 nM T85435 C7T3HJ 44573374 IC50 = 1200 nM T85435 CPMG47 44573375 IC50 = 500 nM T85435 CT1R3Z 44573376 IC50 = 570 nM T85435 CF3N7G 44573377 IC50 = 480 nM T85435 C6BRV7 44573424 IC50 = 310 nM T85435 CXU7T6 44573425 IC50 = 600 nM T85435 C81CVB 44573426 IC50 = 360 nM T85435 CS27CU 44573427 IC50 = 93 nM T85435 CAYJ73 44573467 IC50 = 230 nM T85435 CN6G1U 44573468 IC50 = 400 nM T85435 CO4N5B 44573469 IC50 = 390 nM T85435 CDU34Y 44573502 IC50 = 550 nM T85435 CY81WI 44573503 IC50 = 1100 nM T85435 CM9E7S 44573504 IC50 = 320 nM T85435 C42NEB 44573505 IC50 = 320 nM T85435 CK24OS 44573546 IC50 = 420 nM T85435 C27HSX 44581271 IC50 = 0.8 nM T85435 C53MYT 44588579 IC50 = 320 nM T85435 C6Z3CL 44588719 IC50 = 1800 nM T85435 CXN8P2 44588738 IC50 = 850 nM T85435 CNPI73 44588739 IC50 = 550 nM T85435 CK34PA 44588740 IC50 = 4900 nM T85435 CL67AQ 44588741 IC50 = 235 nM T85435 C6JVC8 44588765 IC50 = 95 nM T85435 C0C9UI 44588766 IC50 > 10000 nM T85435 CT6VG5 44588767 IC50 = 550 nM T85435 CZ1P6B 44588791 IC50 > 10000 nM T85435 C4U8BY 44588793 IC50 = 550 nM T85435 CU6O3G 44588794 IC50 > 10000 nM T85435 C30HRN 44588845 IC50 = 125 nM T85435 CY5T8I 44588846 IC50 > 10000 nM T85435 C5RG0W 44589016 IC50 > 10000 nM T85435 CXE42M 44589045 IC50 > 10000 nM T85435 C5Z3LI 44591740 IC50 > 30000 nM T85435 C9B7LK 44593713 IC50 > 10000 nM T85435 CU3RF1 45139989 IC50 > 10000 nM T85435 CQGZ06 45139991 IC50 > 10000 nM T85435 C4K8BX 45267171 IC50 = 30500 nM T85435 C25VIM 45267176 IC50 = 15600 nM T85435 C7RF4H 45267177 IC50 > 40000 nM T85435 CV94UD 45268038 IC50 = 11900 nM T85435 C64DKR 45268916 IC50 > 40000 nM T85435 CRC85D 45270590 IC50 > 40000 nM T85435 CI82UE 45270897 IC50 = 2300 nM T85435 C36DGY 45272290 IC50 > 40000 nM T85435 COT0W8 45272300 IC50 = 3500 nM T85435 CC79UA 45273165 IC50 = 19800 nM T85435 CNR8G6 45273175 IC50 > 40000 nM T85435 C4UM6Y 45273507 IC50 = 2800 nM T85435 C2C8RH 45379202 IC50 > 100000 nM T85435 C5NB2X 45379203 IC50 > 100000 nM T85435 CT5BJ1 45379204 IC50 > 100000 nM T85435 CB41VP 45379205 IC50 > 100000 nM T85435 C2VUR3 45379340 IC50 > 100000 nM T85435 C8WXT4 45379341 IC50 > 100000 nM T85435 CQL29T 45379342 IC50 > 100000 nM T85435 CM7CB1 45379343 IC50 > 100000 nM T85435 C68WYX 45379344 IC50 > 100000 nM T85435 C27MFU 45379345 IC50 > 100000 nM T85435 C2O6VB 45379346 IC50 = 99000 nM T85435 CLMB07 45379347 IC50 > 100000 nM T85435 C8H5BL 45379490 IC50 = 22000 nM T85435 C4YV6H 45379491 IC50 > 100000 nM T85435 CRK4H3 45379492 IC50 > 100000 nM T85435 CSM20A 45379493 IC50 > 100000 nM T85435 CWP35H 45379494 IC50 > 100000 nM T85435 CV2AZ7 45379495 IC50 > 100000 nM T85435 CMP03L 45379496 IC50 > 100000 nM T85435 C6HM4U 45379605 IC50 > 100000 nM T85435 C6T1SW 45379606 IC50 > 100000 nM T85435 CHNS21 45379607 IC50 = 84000 nM T85435 C8HV1P 45379608 IC50 > 100000 nM T85435 CT6U7X 45379609 IC50 > 100000 nM T85435 C5ATD8 45379610 IC50 > 100000 nM T85435 C2APY4 45379611 IC50 > 100000 nM T85435 CODU08 45379711 IC50 > 100000 nM T85435 C79MTY 45379712 IC50 > 100000 nM T85435 C8LMI5 45379713 IC50 > 100000 nM T85435 CTJQ49 45379714 IC50 > 100000 nM T85435 C15CVY 45379715 IC50 > 100000 nM T85435 CM0P8B 45379716 IC50 > 100000 nM T85435 C9XC4B 45379717 IC50 > 100000 nM T85435 C1U6ST 45379811 IC50 > 100000 nM T85435 CWB1C2 45379812 IC50 > 100000 nM T85435 CATM81 45379814 IC50 > 100000 nM T85435 C4W3OR 45379815 IC50 > 100000 nM T85435 C6E2SC 45482700 IC50 > 10000 nM T85435 CZXH74 45482750 IC50 > 10000 nM T85435 CUA97D 46209401 IC50 > 10000 nM T85435 CZ58FY 46215814 IC50 > 10000 nM T85435 CZBL95 46220496 IC50 = 1808 nM T85435 CKC04F 46220497 IC50 = 35 nM T85435 C92KBM 46229161 IC50 > 100000 nM T85435 CYT37A 46232443 IC50 > 50000 nM T85435 C48ZVW 46232555 IC50 > 50000 nM T85435 CS9B1U 46232556 IC50 > 50000 nM T85435 C7ON5A 46233287 IC50 > 10000 nM T85435 CG24VC 46852202 IC50 = 335 nM T85435 CQL10H 46852353 IC50 = 194 nM T85435 CE3QM1 46869122 IC50 = 369 nM T85435 CLS29B 46872626 IC50 > 10000 nM T85435 CRS61F 46879438 IC50 > 10000 nM T85435 C27JEF 46879439 IC50 = 2628 nM T85435 CF0T8P 46879440 IC50 = 2263 nM T85435 C12RMW 46879441 IC50 = 3486 nM T85435 CH2D7N 46879442 IC50 = 3194 nM T85435 CI6OD8 46879443 IC50 = 1221 nM T85435 C7YD4Q 46879444 IC50 = 1506 nM T85435 C8MN5Q 46879445 IC50 = 1856 nM T85435 CX6SW2 46879446 IC50 = 1092 nM T85435 CNF3V6 46879447 IC50 > 10000 nM T85435 CW46VY 46879448 IC50 = 1365 nM T85435 CLK6X3 46879907 IC50 > 10000 nM T85435 C2A8KO 46880066 IC50 = 1573 nM T85435 CBRP80 46880067 IC50 = 2768 nM T85435 C3FY2B 46880068 IC50 = 3760 nM T85435 CX89TY 46880069 IC50 = 3109 nM T85435 CB0XY1 46880070 IC50 = 4156 nM T85435 CUD81V 46880071 IC50 = 1087 nM T85435 CZP58Q 46880072 IC50 = 1443 nM T85435 CC8OF9 46880073 IC50 > 10000 nM T85435 CF41HG 46880098 IC50 > 10000 nM T85435 C6O2YG 46880099 IC50 = 7121 nM T85435 CI78DM 46880100 IC50 = 29 nM T85435 CU04ZK 46880101 IC50 = 1224 nM T85435 C4E0MF 46880133 IC50 > 10000 nM T85435 COJ16A 46880134 IC50 = 5629 nM T85435 C71MGJ 46880135 IC50 > 10000 nM T85435 C3R6TL 46880213 IC50 = 5435 nM T85435 CT8BQ4 46880214 IC50 = 5935 nM T85435 C0JTO4 46880215 IC50 = 5708 nM T85435 CAFN49 46880216 IC50 > 10000 nM T85435 C6MHP5 46881851 IC50 = 140 nM T85435 C2O8RZ 46886323 IC50 = 80 nM T85435 CW7AR1 46889887 IC50 > 1000 nM T85435 CMNK35 46889911 IC50 > 1000 nM T85435 CHSF07 49806372 IC50 > 1000 nM T85435 C5ME3S 49806721 IC50 = 460 nM T85435 CF91RS 49843531 IC50 > 10000 nM T85435 CE7D2J 49855568 IC50 = 7340 nM T85435 CFD9P3 49855569 IC50 = 1900 nM T85435 C1AU5N 49855758 IC50 = 3700 nM T85435 CIFK93 49855759 IC50 = 1300 nM T85435 CK48OJ 49855760 IC50 = 2500 nM T85435 CZI3M1 49855761 IC50 = 5500 nM T85435 CRPZ58 49855949 IC50 = 2800 nM T85435 CTU0K3 49855950 IC50 = 3000 nM T85435 CF85NL 49855951 IC50 = 7100 nM T85435 CF7YS9 49855952 IC50 = 1400 nM T85435 CJU38G 49855953 IC50 = 1700 nM T85435 C7EAT8 50898348 IC50 = 560 nM T85435 CD2K4R 50908681 IC50 = 622000 nM T85435 C2Y6QS 50938552 IC50 > 10000 nM T85435 CP7B9V 50942696 IC50 = 1380 nM T85435 CH4G3V 51000498 IC50 = 153 nM T85435 C9NYP4 51036677 IC50 > 10000 nM T85435 C4WRY3 51037112 IC50 > 10000 nM T85435 CRI28Z 51037948 IC50 > 10000 nM T85435 CEQN27 52936621 Ki > 1000 nM T85435 CW09EM 52945447 IC50 = 380 nM T85435 CNV67T 52945448 IC50 = 1600 nM T85435 C30RAL 52946684 IC50 = 9900 nM T85435 C1FIW8 53315285 IC50 = 12 nM T85435 CF20TR 53317353 IC50 = 504 nM T85435 C8QL7R 53317354 IC50 = 62 nM T85435 C5QFO0 53317399 IC50 = 20 nM T85435 C6E9AG 53317400 IC50 = 550 nM T85435 C8UY3B 53317401 IC50 = 2300 nM T85435 CMDP24 53317655 IC50 > 3000 nM T85435 C5M3OC 53318635 IC50 = 2694 nM T85435 C6Q8MV 53318636 IC50 > 3000 nM T85435 CTG1Z2 53318637 IC50 = 573 nM T85435 CGX38E 53318663 IC50 = 334 nM T85435 C2GQS5 53318695 IC50 > 3000 nM T85435 CXK28V 53318696 IC50 = 1400 nM T85435 CP2ZE6 53318802 IC50 = 1150 nM T85435 CM0L9V 53319073 IC50 = 351 nM T85435 CJ2D3F 53319267 IC50 = 76 nM T85435 C5DUO3 53319892 IC50 = 48 nM T85435 CA4I8S 53319963 IC50 = 1860 nM T85435 CR7S3Q 53320012 IC50 = 370 nM T85435 C24TVU 53321197 IC50 = 700 nM T85435 C5B2LC 53321198 IC50 = 260 nM T85435 CK7A8Y 53321265 IC50 > 10000 nM T85435 C9D8EB 53321266 IC50 = 233 nM T85435 C20IVP 53321284 IC50 = 11 nM T85435 CC63UD 53321285 IC50 = 30 nM T85435 CMC30H 53321320 IC50 = 800 nM T85435 C09SRW 53321321 IC50 = 500 nM T85435 CNT53F 53321676 IC50 = 820 nM T85435 CQD92F 53322588 IC50 = 189 nM T85435 CYX1F2 53322608 IC50 = 404 nM T85435 CE27TP 53323941 IC50 = 34 nM T85435 C2TCM1 53323942 IC50 = 231 nM T85435 C54YZQ 53323973 IC50 = 1200 nM T85435 C2W9OA 53324451 IC50 > 10000 nM T85435 C3DO4U 53325211 IC50 > 10000 nM T85435 C0XD5M 53325268 IC50 > 10000 nM T85435 C9UB7N 53325269 IC50 = 230 nM T85435 CSU20C 53325270 IC50 = 300 nM T85435 C4YG5H 53325271 IC50 = 930 nM T85435 CXOL24 53325517 IC50 > 6500 nM T85435 CO57DC 53325540 IC50 = 200 nM T85435 CEK97L 53325637 IC50 = 320 nM T85435 CI41VZ 53326513 IC50 = 8 nM T85435 CWL68I 53326881 IC50 = 490 nM T85435 CNPM14 53341082 IC50 > 3000 nM T85435 C0SWH5 53348216 IC50 > 40000 nM T85435 C8ZRE3 53356518 IC50 = 9142 nM T85435 CM7P3W 53357328 IC50 = 310 nM T85435 C4QO8D 53364164 IC50 > 40000 nM T85435 CK52GI 53380818 IC50 = 9 nM T85435 C8NA4L 53384644 IC50 > 30000 nM T85435 C24FQU 53465297 IC50 = 1137 nM T85435 C67XFO 53482132 IC50 = 1400 nM T85435 CI12VS 54577678 IC50 = 19 nM T85435 COF6B0 54577892 IC50 = 123 nM T85435 C5TAL7 54577893 IC50 = 326 nM T85435 CPS75F 54577894 IC50 > 2000 nM T85435 C17PKQ 54577895 IC50 = 1874 nM T85435 C2ECL9 54577896 IC50 = 366 nM T85435 CZ9W6N 54577897 IC50 = 391 nM T85435 C08ABD 54578104 IC50 = 206 nM T85435 CIV58E 54578105 IC50 = 160 nM T85435 C0W4QA 54578108 IC50 = 934 nM T85435 C0KI7N 54578323 IC50 = 1171 nM T85435 COEX71 54578324 IC50 = 809 nM T85435 CE1ZK6 54759168 IC50 > 10000 nM T85435 C1XS2J 54760383 IC50 > 10000 nM T85435 C69FXM 54760600 IC50 = 6499 nM T85435 C9EMO2 54765177 IC50 = 1290 nM T85435 CK9JO3 56597774 IC50 = 3111 nM T85435 C8AZB0 56597931 IC50 = 886 nM T85435 CM8JX1 56604907 IC50 = 10 nM T85435 CN9QD7 56643097 IC50 > 10000 nM T85435 CGZ76M 56658177 IC50 = 266 nM T85435 C9RO7H 56659710 IC50 = 150 nM T85435 CQX1B0 56659754 IC50 > 40000 nM T85435 CPEQ43 56659755 IC50 > 40000 nM T85435 CM15EG 56659756 IC50 > 40000 nM T85435 COT59W 56659757 IC50 > 40000 nM T85435 C9JN5I 56659776 IC50 > 40000 nM T85435 CO6XJ2 56659777 IC50 > 40000 nM T85435 CO7N3J 56659778 IC50 > 40000 nM T85435 CR2AZ4 56659779 IC50 > 40000 nM T85435 CP02ZN 56663035 IC50 > 40000 nM T85435 C0TA4N 56663131 IC50 > 40000 nM T85435 C10HLV 56663132 IC50 > 40000 nM T85435 C8CRO9 56663133 IC50 > 40000 nM T85435 CVL35R 56663134 IC50 > 40000 nM T85435 C4AJE2 56663169 IC50 = 180 nM T85435 C3ZXK9 56663170 IC50 = 6300 nM T85435 C3R4VA 56663171 IC50 = 740 nM T85435 C28VGO 56663172 IC50 = 710 nM T85435 C0BKE4 56663174 IC50 = 430 nM T85435 CC6Y5B 56663231 IC50 > 40000 nM T85435 CTPK64 56663250 IC50 > 40000 nM T85435 CWYO21 56663251 IC50 > 40000 nM T85435 CFMW78 56663252 IC50 > 40000 nM T85435 CP07FJ 56665099 IC50 = 357 nM T85435 C0NCP7 56666587 IC50 > 40000 nM T85435 C8XZ4O 56666620 IC50 = 840 nM T85435 CI9CK1 56666661 IC50 > 40000 nM T85435 CKBD90 56666683 IC50 > 40000 nM T85435 C0Q4XE 56666684 IC50 > 40000 nM T85435 CEH31Y 56668417 IC50 = 295 nM T85435 C9DJH8 56670079 IC50 > 40000 nM T85435 C46PYQ 56670080 IC50 > 40000 nM T85435 C37WLX 56670081 IC50 > 40000 nM T85435 CB83JE 56670082 IC50 > 40000 nM T85435 C8A4RP 56670104 IC50 > 40000 nM T85435 CC54FO 56670105 IC50 > 40000 nM T85435 C9OA3E 56673602 IC50 > 40000 nM T85435 C59WKG 56673603 IC50 > 40000 nM T85435 C4HKA0 56673622 IC50 > 40000 nM T85435 C9TH6I 56673623 IC50 > 40000 nM T85435 CSZ9P6 56676866 IC50 = 1700 nM T85435 CMO45E 56676867 IC50 = 540 nM T85435 CLMK58 56676868 IC50 = 930 nM T85435 C07DET 56676869 IC50 = 460 nM T85435 CFC14P 56676919 IC50 > 40000 nM T85435 CXQ3W5 56676939 IC50 > 40000 nM T85435 CS92FR 56676940 IC50 > 40000 nM T85435 C87OYI 56676941 IC50 > 40000 nM T85435 C4ZRM2 56678466 IC50 = 840 nM T85435 C4RJ5H 56680184 IC50 = 920 nM T85435 C8GT6K 56680185 IC50 = 77 nM T85435 C4ARS6 56680232 IC50 > 40000 nM T85435 C7XH1J 56680233 IC50 > 40000 nM T85435 CE8N6R 56680259 IC50 > 40000 nM T85435 CO21ZG 56680260 IC50 > 40000 nM T85435 C86EIX 56680261 IC50 > 40000 nM T85435 C45RZV 56683336 IC50 = 150 nM T85435 CN5W3I 56683485 IC50 > 40000 nM T85435 C8ZJE5 56683588 IC50 > 40000 nM T85435 C5UKI1 56683589 IC50 > 40000 nM T85435 C7Y2EO 56683590 IC50 > 40000 nM T85435 CUT2G8 56835062 IC50 = 380 nM T85435 CI5ZJ7 56835161 IC50 > 100000 nM T85435 CN1A8C 56945612 IC50 = 222 nM T85435 CGW9B2 56945613 IC50 = 149 nM T85435 CE95CG 56945614 IC50 = 164 nM T85435 CA3U2R 56945615 IC50 = 579 nM T85435 C6AJC0 56945727 IC50 = 161 nM T85435 C5FY9U 56945728 IC50 = 222 nM T85435 C2OS1K 56945729 IC50 = 2967 nM T85435 CWS36I 56945730 IC50 = 747 nM T85435 CY39NF 56945731 IC50 > 10000 nM T85435 CNS43L 56945844 IC50 = 410 nM T85435 CF0X2H 56945845 IC50 = 552 nM T85435 CAK91L 56955954 IC50 > 3600 nM T85435 CF5JV6 56966833 IC50 = 90.6 nM T85435 C1WJT2 56966906 IC50 = 1179 nM T85435 C26MCX 56966977 IC50 = 702 nM T85435 CX34KP 56966978 IC50 = 57.2 nM T85435 CDS06V 56973548 IC50 = 5011.87 nM T85435 CUAV97 56973549 IC50 = 7943.28 nM T85435 CI0K7Y 56973550 IC50 = 2511.89 nM T85435 CPHX64 57325478 IC50 > 50000 nM T85435 CQ9BW4 57325479 IC50 > 50000 nM T85435 CDW6R2 57329726 IC50 = 536 nM T85435 CM3G0E 57390177 IC50 = 2999 nM T85435 C0TM9U 57390203 IC50 = 473 nM T85435 C1UZE5 57390692 IC50 = 16000 nM T85435 C2ZKN5 57390751 IC50 = 41 nM T85435 CGJN96 57390792 IC50 = 5.2 nM T85435 CONV59 57390937 IC50 = 210 nM T85435 C9OGW0 57391592 IC50 = 80 nM T85435 CS6FV1 57391593 IC50 = 130 nM T85435 C31NML 57391953 IC50 = 598 nM T85435 CDF6J2 57392000 IC50 = 1729 nM T85435 CWB09F 57392558 IC50 = 120 nM T85435 CNR9I1 57392730 IC50 = 93 nM T85435 C0BAR8 57392731 IC50 = 120 nM T85435 CB0C7T 57392732 IC50 = 53 nM T85435 C2PJN1 57393680 IC50 = 583 nM T85435 CRO72U 57393705 IC50 = 71 nM T85435 CDTX78 57394203 IC50 = 26 nM T85435 C3VNY5 57394377 IC50 = 428 nM T85435 CPZH71 57395063 IC50 = 12 nM T85435 CX7A9P 57395064 IC50 = 32 nM T85435 C4QER2 57395065 IC50 = 50 nM T85435 CD0F8J 57395066 IC50 = 34 nM T85435 C8W6IG 57395117 IC50 > 30000 nM T85435 CK1D4R 57395398 IC50 = 1807 nM T85435 CV8OD3 57395399 IC50 = 273 nM T85435 CG2I4M 57395970 IC50 = 13 nM T85435 CD0OQ4 57396144 IC50 > 10000 nM T85435 CE1WT0 57396145 IC50 = 1415 nM T85435 C3AW8K 57396220 IC50 = 42 nM T85435 C0Z9RG 57396834 IC50 = 7.5 nM T85435 CXA2O5 57396835 IC50 = 6 nM T85435 CB13SR 57396836 IC50 = 40 nM T85435 CD7KN4 57396837 IC50 = 42 nM T85435 CL8G3R 57397237 IC50 = 945 nM T85435 CUR52C 57397767 IC50 = 42 nM T85435 C9BUV4 57397962 IC50 > 1000 nM T85435 C6HJ1A 57397963 IC50 > 10000 nM T85435 CILC36 57398016 IC50 = 180 nM T85435 CUR70J 57398017 IC50 = 90 nM T85435 CEV41G 57398592 IC50 = 10 nM T85435 CRSL84 57398926 IC50 = 2999 nM T85435 C0J2UD 57399430 IC50 = 40 nM T85435 CJ30GQ 57399673 IC50 = 210 nM T85435 COU36H 57399674 IC50 = 52 nM T85435 CU3MV1 57401430 IC50 = 52 nM T85435 CMZ7B1 57401431 IC50 = 80 nM T85435 CJP2L1 57401432 IC50 = 80 nM T85435 CZ5VR8 57402451 IC50 = 370 nM T85435 CJF86Y 57402453 IC50 = 3211 nM T85435 CGE8I2 57403115 IC50 = 9124 nM T85435 C8P6RD 57505528 IC50 > 10000 nM T85435 CVK0G4 58056356 IC50 > 50000 nM T85435 C4V7FY 58191950 IC50 = 41000 nM T85435 CPCA29 58191961 IC50 = 65000 nM T85435 C7HF1L 58191965 IC50 = 36000 nM T85435 C8LWY9 58191997 IC50 = 150000 nM T85435 CTWG72 58290872 IC50 = 416 nM T85435 C24BEZ 59577331 IC50 = 457 nM T85435 C1JCV8 59577340 IC50 = 823 nM T85435 CT3J2N 59577341 IC50 = 353 nM T85435 C1CSH0 59577345 IC50 = 1642 nM T85435 CJZ71Q 59577355 IC50 = 906 nM T85435 CIB62O 59577356 IC50 = 653 nM T85435 C75VNB 59577361 IC50 = 1489 nM T85435 C7QY2B 59577365 IC50 = 196 nM T85435 CXJ63M 59603829 IC50 > 100000 nM T85435 CQEU96 59603842 IC50 > 10000 nM T85435 CPU2E3 59737752 IC50 = 414 nM T85435 CF8E1J 59764390 IC50 = 564 nM T85435 CC48EN 59764418 IC50 = 281.8 nM T85435 C4NBG7 59764433 IC50 = 510 nM T85435 C40UZT 59764460 IC50 = 326.5 nM T85435 C6AQX8 59764524 IC50 = 464 nM T85435 C5B0JN 59764577 IC50 = 1186 nM T85435 C1MR8Q 60097495 IC50 > 1000 nM T85435 COM48T 60154284 IC50 = 3162.28 nM T85435 CB7KE0 60154285 IC50 = 7943.28 nM T85435 CO75BK 60154286 IC50 = 3981.07 nM T85435 CEF48W 60154326 IC50 = 630.96 nM T85435 CSZA16 60155724 IC50 > 3600 nM T85435 CK6WO0 66552478 IC50 < 10000 nM T85435 CY0C3J 66829998 IC50 > 10000 nM T85435 C82YDV 66830004 IC50 = 215 nM T85435 CMN68E 66830116 IC50 = 12 nM T85435 CX7LS6 66830288 IC50 = 71 nM T85435 CY31IS 66830367 IC50 = 2012 nM T85435 COH5N4 66830485 IC50 = 32 nM T85435 CBU5X6 66830555 IC50 = 247 nM T85435 CRH43K 66830651 IC50 = 37 nM T85435 C2ZEX1 66929146 EC50 = 2750 nM T85435 C1HSE0 67035086 IC50 = 638 nM T85435 CWI6K5 67035106 IC50 = 471 nM T85435 C38RGB 67035556 IC50 = 930 nM T85435 CV3HW2 67035568 IC50 = 100 nM T85435 CK80LJ 67130050 IC50 > 10000 nM T85435 CV63UL 67240318 IC50 > 10000 nM T85435 CDE47U 67264047 IC50 = 1301 nM T85435 C7BF3N 67264510 IC50 = 89 nM T85435 CEV60X 68156947 IC50 = 9.9 nM T85435 C59RQC 68165302 IC50 = 314 nM T85435 CL97JB 68165311 IC50 = 399 nM T85435 CM1ZC3 68165315 IC50 = 284 nM T85435 CET2P8 68165322 IC50 = 285 nM T85435 C61QGN 68165327 IC50 = 489 nM T85435 CFRK82 68165328 IC50 = 4.7 nM T85435 CLH97K 68165338 IC50 = 1683 nM T85435 C7Y8KG 68165350 IC50 = 171 nM T85435 C2AX3V 68165354 IC50 = 162 nM T85435 C2B3TL 68165357 IC50 = 483 nM T85435 C81YOZ 68165362 IC50 = 343 nM T85435 CLGN08 68165375 IC50 = 14.1 nM T85435 C82RIW 68165380 IC50 = 253 nM T85435 CH5Y2P 68165382 IC50 = 339 nM T85435 C3H5XQ 68165389 IC50 = 130 nM T85435 C0WFX2 68165395 IC50 = 0.88 nM T85435 C0G7QF 68165398 IC50 = 700 nM T85435 CNK7S3 68165399 IC50 = 103 nM T85435 C78BZG 68165403 IC50 = 85.3 nM T85435 CZ1Q8W 68165412 IC50 = 55.2 nM T85435 CYD2V8 68165414 IC50 = 171 nM T85435 CVGJ74 68165424 IC50 = 13.7 nM T85435 CN27QC 68165467 IC50 = 367 nM T85435 CO2LF9 68166178 IC50 = 270 nM T85435 CR1U7L 68166323 IC50 = 397 nM T85435 C4VQJ8 68166330 IC50 = 459 nM T85435 C8I7GC 68293638 IC50 = 166 nM T85435 CD56XK 68293660 IC50 = 36 nM T85435 C7GRV2 68755406 IC50 = 3480 nM T85435 CLY7I4 68971880 EC50 = 5030 nM T85435 CM4WN5 68976126 EC50 = 1800 nM T85435 C5DGR9 69036886 IC50 = 1192 nM T85435 C2S8YO 69270579 EC50 = 300 nM T85435 CMPQ52 69271243 EC50 = 4760 nM T85435 CB13CE 69272823 EC50 = 1320 nM T85435 CC90HU 70684001 IC50 = 319 nM T85435 CB1X4E 70696546 IC50 = 91 nM T85435 CH0B8N 70789756 IC50 > 30000 nM T85435 CEBO91 71452977 IC50 > 10000 nM T85435 CCN01X 71547862 IC50 > 10000 nM T85435 CA3O6K 71552696 IC50 = 4650 nM T85435 C1NPL0 71552941 IC50 > 30000 nM T85435 CA4PS8 71552942 IC50 > 30000 nM T85435 C3UA9C 71553011 IC50 = 30000 nM T85435 CEZ15Y 71553012 IC50 = 18620 nM T85435 CVIA91 71553085 IC50 = 30000 nM T85435 C1TR3O 71553152 IC50 = 30000 nM T85435 CZ31PU 71583657 IC50 > 10000 nM T85435 C72KYC 71763639 IC50 = 784 nM T85435 C8ZY1V 71763864 IC50 = 1920 nM T85435 C19WUN 71764054 IC50 = 541.5 nM T85435 C56IPY 71764055 IC50 = 197.2 nM T85435 CG5S3Y 71764056 IC50 = 344.5 nM T85435 CS8BR1 71764218 IC50 = 240.1 nM T85435 CNW35A 71764219 IC50 = 4874 nM T85435 CS6DN3 71764394 IC50 = 891.5 nM T85435 CUGC68 71764395 IC50 = 361.1 nM T85435 C2NJ4Z 71764396 IC50 = 401 nM T85435 CGWT31 71764397 IC50 = 1643 nM T85435 C0KNW2 71764604 IC50 = 418 nM T85435 CX75YR 73352604 IC50 = 158.49 nM T85435 CQZ0L8 78158242 IC50 = 129 nM T85435 CQ9H4U 86277844 IC50 = 5700 nM T85435 C0QK9F 86288869 IC50 = 2872 nM T85435 CPG3A5 86302574 IC50 > 30000 nM T85435 C9NTP1 86677234 IC50 = 21 nM T85435 C58VLT 89726147 IC50 = 79 nM T85435 CA49UY 89726151 IC50 = 68 nM T85435 C1HW4B 89735655 IC50 > 100000 nM T85435 CY6K5P 89738540 IC50 = 348 nM T85435 CIXB02 89738547 IC50 = 129 nM T85435 CH58TV 89773144 IC50 = 1684 nM T85435 CSX63K 89773146 IC50 = 26 nM T85435 CTV2C7 89774514 IC50 = 270 nM T85435 CY0UC4 90645194 IC50 > 10000 nM T85435 C0S1HF 90655767 IC50 = 170 nM T85435 CW5ZR6 90655768 IC50 = 39 nM T85435 C51MOA 90655769 IC50 > 12500 nM T85435 CZ6U5W 90655770 IC50 > 12500 nM T85435 C7P6FQ 90655771 IC50 = 7867 nM T85435 CXA18Y 90655772 IC50 = 5228 nM T85435 C15GJU 90655773 IC50 = 11805 nM T85435 C25CWH 90655774 IC50 > 12500 nM T85435 CFRI21 90655775 IC50 > 12500 nM T85435 CAIL45 90655776 IC50 > 12500 nM T85435 CVYA67 90655777 IC50 > 12500 nM T85435 C4GU0L 90665978 IC50 = 1919 nM T85435 CP65IG 90665979 IC50 > 3000 nM T85435 CZA0F4 90665980 IC50 = 253 nM T85435 CJF1Z9 90665981 IC50 = 787 nM T85435 CY90XF 90665982 IC50 = 901 nM T85435 CR1Q9I 90665983 IC50 = 158 nM T85435 CV62FB 90665984 IC50 = 1013 nM T85435 C8EUC3 90665985 IC50 = 510 nM T85435 CXEJ32 90665986 IC50 = 169 nM T85435 CDQ56W 90665987 IC50 = 54 nM T85435 C5E2FJ 90665988 IC50 = 48 nM T85435 C4TPN8 90665989 IC50 = 24 nM T85435 CBG6E7 91885506 IC50 = 81 nM T85435 C0Y8ZK 91933875 IC50 > 1000 nM T85435 C05NTY 101884761 IC50 = 35 nM T85435 CWM71R 101884762 IC50 = 9 nM T85435 CN0EF8 117929515 IC50 = 110 nM T85435 C3N5IY 117955447 IC50 = 736 nM T85435 C4CH7J 117955548 IC50 = 71 nM T85435 C5T4WU 117955577 IC50 = 1763 nM T85435 C2T4MB 117955613 IC50 = 915 nM T85435 C07ACT 117955744 IC50 = 814 nM T85435 C5K2DA 117955863 IC50 = 722 nM T85435 C50ANY 117955890 IC50 > 2000 nM T85435 CY7BI2 118706214 IC50 > 10000 nM T85435 C3KLI5 118723185 IC50 > 100000 nM T85435 C08KEM 122179540 IC50 = 8600 nM T85435 C3AJ4C 122179546 IC50 = 8800 nM T85435 CG0RP7 122179547 IC50 = 5300 nM T85435 C1A0SQ 122179548 IC50 = 6000 nM T85435 CND7S8 122186934 IC50 = 25 nM T85435 CUBD36 122186935 IC50 = 21 nM T85435 CP65NK 122186936 IC50 = 11 nM T85435 CA74DF 122186937 IC50 = 5.2 nM T85435 CK8G1M 122186938 IC50 = 5.1 nM T85435 CCR3P8 122186939 IC50 = 2 nM T85435 CQW9Z5 122186940 IC50 = 12 nM T85435 CSEJ41 127048207 IC50 = 189 nM T85435 CDK3C6 127049147 IC50 = 128 nM T85435 C2MF9I 127049148 IC50 = 3.4 nM T85435 CV1E5D 127049149 IC50 = 6.05 nM T85435 C07TZN 127049440 IC50 = 8.44 nM T85435 C2FE1A 127049463 IC50 = 2.16 nM T85435 C7ODG2 127049464 IC50 = 43.2 nM T85435 C7A4OJ 127049465 IC50 = 5.1 nM T85435 C4WKQ5 127052926 IC50 = 1163 nM T85435 CHQJ02 127052979 IC50 = 81.7 nM T85435 C9CVB0 129048532 IC50 = 14 nM T85435 CO1ST8 129065476 IC50 = 2.8 nM T85435 CXN46D 129148000 IC50 = 2.2 nM T85435 C97GOL 129896918 IC50 = 6 nM T85435 CUO0C5 132156633 IC50 > 10000 nM T85435 C1WO9J 134132421 IC50 = 103 nM T85435 CW04KZ 134141466 IC50 = 145 nM T85435 CAL5D8 134145302 IC50 = 435 nM T85435 CQU86Z 134146557 IC50 = 994 nM T85435 CFG60Q 134148895 IC50 = 382 nM T85435 C9Z1VM 134153244 IC50 = 403 nM T85435 C7H8GQ 134157229 IC50 = 508 nM T85435 CK5VG4 134219752 IC50 = 11 nM T85435 C2AN7T 134611886 IC50 > 100000 nM T85435 CU60YC 135431661 IC50 > 30000 nM T85435 C16XLU 135454992 IC50 = 550 nM T85435 C64EMD 135500075 IC50 > 10000 nM T85435 CVZ08D 135509841 IC50 = 4000 nM T85435 CJI0G1 135520135 IC50 > 10000 nM T85435 CTJ48K 135524085 IC50 = 7800 nM T85435 CUT1W7 135524168 IC50 > 10000 nM T85435 CX4ZB3 135863110 IC50 > 10000 nM T85435 CF48JM 135908497 IC50 > 100000 nM T85435 C3YO9W 135929504 IC50 > 100000 nM T85435 C1NH5A 135929506 IC50 > 100000 nM T85435 CA8UN4 135929507 IC50 > 100000 nM T85435 C7J9ZD 135929508 IC50 > 100000 nM T85435 CB2P3H 135929509 IC50 > 100000 nM T85435 CJ1S7B 135929510 IC50 > 100000 nM T85435 C4IMU5 135929525 IC50 = 11000 nM T85435 C65NTO 135929526 IC50 > 100000 nM T85435 CAV34T 135929527 IC50 > 100000 nM T85435 C9EX0T 135929541 IC50 > 100000 nM T85435 CE4OU5 135929542 IC50 > 100000 nM T85435 CIPA79 135937899 IC50 > 10000 nM T85435 C6H0AI 135957039 IC50 > 10000 nM T85435 CHA4N2 136013680 IC50 > 10 nM T85435 CBS87V 136016385 IC50 = 7080 nM T85435 C05IWG 136016386 IC50 = 9330 nM T85435 COPL16 136016393 IC50 = 5750 nM T85435 CUP47N 136016409 IC50 = 5010 nM T85435 C4RMV8 136016410 IC50 = 20000 nM T85435 C48DLS 136123445 IC50 = 51 nM T85435 CH64ID 136175114 IC50 > 10000 nM T85435 C1YUD0 136219394 IC50 > 10 nM T85435 CIU8W3 136254389 IC50 > 10 nM T85435 CSGM03 137210056 IC50 > 10000 nM T85435 C25ERN 137631967 IC50 = 431.2 nM T85435 CORJ86 137632190 EC50 = 4580 nM T85435 CI1E8V 137634241 IC50 = 2130 nM T85435 CMN0V1 137634592 IC50 = 300 nM T85435 CH7Z2E 137636265 IC50 = 7.5 nM T85435 C5T0YN 137636330 EC50 > 10000 nM T85435 C06JRX 137637094 IC50 = 417.5 nM T85435 C2ZXS7 137640634 IC50 = 260 nM T85435 CJ5AV0 137641991 EC50 = 1005 nM T85435 CE2WN1 137648666 IC50 = 21 nM T85435 C1DK0P 137651391 IC50 = 887.6 nM T85435 C5F7TG 137654160 IC50 = 130 nM T85435 CJC62Q 137655585 IC50 = 2.1 nM T85435 CV5H3Z 137657932 IC50 = 91.6 nM T85435 C0B7RX 137658642 IC50 > 10000 nM T85435 C6VB3O 145925651 IC50 >= 5000 nM T85435 CW3RV1 145953992 IC50 > 10000 nM T85435 CCL34O 145954234 IC50 = 1258.93 nM T85435 C4ZH8E 145954241 IC50 > 10000 nM T85435 CNT8O5 145954713 IC50 = 3981.07 nM T85435 CB0F7N 145955167 IC50 = 3162.28 nM T85435 CJDG56 145960632 IC50 > 10000 nM T85435 CB7TW3 145960672 IC50 = 1258.93 nM T85435 CH6G1S 145960935 IC50 = 1258.93 nM T85435 C6ZJQ4 145961055 IC50 = 3162.28 nM T85435 CE21QP 145961382 IC50 > 10000 nM T85435 CQ9FN7 145961544 IC50 = 794.33 nM T85435 C23GXR 145961663 IC50 = 316.23 nM T85435 CJ0K8Z 145962062 IC50 = 3981.07 nM T85435 CV0T1U 145962184 IC50 = 316.23 nM T85435 CA2RO4 145962531 IC50 = 398.11 nM T85435 CCL79I 145963000 IC50 = 158.49 nM T85435 CI0V8W 145963248 IC50 > 10000 nM T85435 C0JX1P 145963398 IC50 > 10000 nM T85435 CJZ4G3 145963549 IC50 = 630.96 nM T85435 C9V6AQ 145963687 IC50 = 1584.89 nM T85435 C2MD1Q 155513187 IC50 > 10000 nM T85435 CCFN07 155525418 EC50 = 4.01 nM T85435 C78MZC 155536330 IC50 = 8 nM T85435 CE46SL 155540854 IC50 > 30000 nM T85435 C5O4JM 155540856 IC50 = 9790 nM T85435 CGVU70 155554426 IC50 > 30000 nM T85435 D00EMH 56597775 IC50 = 1418 nM T85435 D00ERW 44444843 Ki > 5238 nM T85435 D00HVA 11624601 Ki > 5200 nM T85435 D02BXJ 46864270 IC50 > 3000 nM T85435 D02NNT 53232451 IC50 > 10000 nM T85435 D02XHC 448912 IC50 = 60000 nM T85435 D03DZO 11715767 IC50 > 10000 nM T85435 D04NGS 5330790 IC50 > 100000 nM T85435 D04PEI 11467730 IC50 = 1100 nM T85435 D04ZWF 53396311 IC50 > 2000 nM T85435 D06HVH 54613583 IC50 > 10000 nM T85435 D06PJW 25182616 IC50 = 79 nM T85435 D06QWO 14824655 IC50 > 10 ug.mL-1 T85435 D07ADX 54764565 IC50 = 200 nM T85435 D07OAT 456214 IC50 = 5000 nM T85435 D07OCA 5330812 IC50 > 10000 nM T85435 D08HFG 24809764 IC50 > 10000 nM T85435 D09HVH 135566652 IC50 > 10 nM T85435 D09PTP 57325421 IC50 = 662 nM T85435 D09RYV 9911652 IC50 = 71000000 nM T85435 D0A1CM 5281855 IC50 = 340 nM T85435 D0C2GE 67161540 IC50 = 4100 nM T85435 D0G3SZ 6918469 IC50 = 5.6 ug.mL-1 T85435 D0G4CS 25229528 IC50 = 597 nM T85435 D0L7MM 43680262 IC50 = 5150 nM T85435 D0M4SY 135440466 IC50 = 73 nM T85435 D0O6OH 71553154 IC50 = 6180 nM T85435 D0Q3GG 667601 IC50 = 640000 nM T85435 D0Q3NG 11715520 Ki > 5200 nM T85435 D0R2WK 16038120 IC50 = 43.7 nM T85435 D0RO9R 50942314 IC50 = 730 nM T85435 D0S7IE 11658882 Ki > 5200 nM T85435 D0T3PW 5281672 Ki = 2600 nM T85435 D0T8NU 16757525 IC50 > 4000 nM T85435 D0W9KO 43743432 IC50 = 2250 nM T85435 D0YE1X 9927943 IC50 > 100000 nM T85435 D0YZ7H 9797370 IC50 > 100000 nM T77365 D04JEE 4946 EC50 > 5011.87 nM T77365 D04OSE 4485 Ki = 22200 nM T77365 D06IAR 60961 Ki = 20 nM T77365 D09AMZ 1676 EC50 = 7200 nM T77365 D0B3HD 2519 Ki = 2480 nM T77365 D0F8RA 2153 Ki = 0.6 nM T77365 D0I0RJ 16231 Ki = 3280 nM T77365 D0R4UW 449193 IC50 > 1000 nM T77365 D0XE1C 219024 Ki = 290 nM T77365 D0Z7ZM 135398744 Ki = 199.53 nM T77365 D00OAU 9869857 IC50 = 0.4 nM T77365 D00SUK 216466 Ki = 6400 nM T77365 D02YQO 10668061 Ki = 0.048 nM T77365 D03OQI 11618368 Ki = 0.3 nM T77365 D06MIQ 9910098 Ki = 58.5 nM T77365 D07TEP 10117987 Ki = 0.5 nM T77365 D09TFB 9896267 IC50 = 4400 nM T77365 D0D5VJ 9833519 Ki = 4 nM T77365 D0F4ZY 5311037 Ki = 2.2 nM T77365 D0F5UN 9953065 Ki = 398 nM T77365 D0FD6D 11751922 Ki = 500 nM T77365 D0G4CF 11270783 Ki = 3280 nM T77365 D0L5VS 6448585 IC50 = 1 nM T77365 D0LI1C 44469321 IC50 > 30000 nM T77365 D0M3IN 1188 EC50 > 100000 nM T77365 D0QG9A 9805430 Ki = 0.5 nM T77365 D0U0KR 3035850 Ki = 401 nM T77365 D0W9NO 146207 Ki = 31.8 nM T77365 D0X0IY 64627 Ki = 108 nM T77365 D0Y6ZK 123683 Ki = 32 nM T77365 D0Z3PO 21874557 Ki = 1.3 nM T77365 D0Z9RJ 11561692 Ki > 10000 nM T77365 D08ECB 11716665 Ki > 2500 nM T77365 D0I5VA 11248240 Ki = 2300 nM T77365 D0CH7Z 128784 Ki = 2100 nM T77365 D00YSJ 158795 Ki = 2315 nM T77365 D01VPK 6439091 Ki = 1300 nM T77365 D07ESH 176408 Ki = 0.6 nM T77365 D0J2UW 3086599 EC50 = 2.12 nM T77365 D0NQ5I 65710 Ki = 760 nM T77365 D0V5DX 9884817 Ki = 1330 nM T77365 D0Y6GJ 176407 Ki = 0.1 nM T77365 C7B8VJ 44405080 Ki = 3250 nM T77365 CF92BM 45482610 Ki = 3250 nM T77365 C6GN7M 40692 Ki = 6553 nM T77365 CY8K9D 70639 EC50 > 100000 nM T77365 CKF52M 71593 Ki > 100000 nM T77365 CA9Z0E 78268 Ki = 115 nM T77365 C3SPQ5 95121 Ki > 100000 nM T77365 C2CG8M 98567 Ki = 466 nM T77365 CMT4D5 104924 Ki = 51.3 nM T77365 C57IVM 126054 Ki = 370 nM T77365 C6OGM1 131432 Ki = 9.3 nM T77365 C2J0SC 131450 Ki = 579 nM T77365 CU7A5O 149362 EC50 = 12 nM T77365 C5N6TM 161713 EC50 = 600 nM T77365 CEG2T8 169316 EC50 = 1300 nM T77365 CF59MP 169662 EC50 = 5400 nM T77365 CN1V0P 174907 EC50 = 9600 nM T77365 CL08HI 185566 Ki = 30000 nM T77365 CA6E5H 215492 Ki = 505 nM T77365 CD0MT5 215610 EC50 = 225 nM T77365 C0Y8GT 218667 EC50 = 8300 nM T77365 CT58VJ 236871 Ki = 640 nM T77365 CMH1F9 308531 Ki = 381 nM T77365 C5BK1O 314836 Ki > 10000 nM T77365 CYU2W7 340706 Ki = 1300 nM T77365 C7QO3K 343627 EC50 = 10600 nM T77365 C9GV7U 350737 EC50 = 69200 nM T77365 CVD90Q 377427 Ki = 2000 nM T77365 CLZE79 386674 Ki > 10000 nM T77365 CW4FT7 395949 Ki = 79.43 nM T77365 C58QWF 456309 Ki = 61 nM T77365 C8EDA0 500900 Ki = 3420 nM T77365 CYE04Q 541615 Ki = 169.82 nM T77365 C9GZ0J 541903 Ki = 2370 nM T77365 CI0CW2 570244 Ki = 400 nM T77365 CE9CN4 571407 Ki = 224 nM T77365 C2Y4TD 577307 Ki = 220 nM T77365 C5B6GT 591132 Ki > 100000 nM T77365 CX31PR 621302 Ki = 4900 nM T77365 CSV78R 626711 Ki = 59100 nM T77365 CQ4M6T 631000 Ki = 2700 nM T77365 CA9Y0C 648481 Ki = 707.95 nM T77365 CO3ZC7 677535 Ki = 700 nM T77365 C03TBX 679358 Ki > 100000 nM T77365 CT3NQ1 684194 Ki = 232 nM T77365 C2HTM9 686655 Ki = 106 nM T77365 C5FEO8 700373 Ki = 31000 nM T77365 CW6K7C 706959 Ki = 9100 nM T77365 CJ5A4P 707926 Ki = 1995.26 nM T77365 C5X7WA 711464 Ki = 201 nM T77365 CJN2G4 714281 Ki = 1600 nM T77365 CUV5M3 715162 Ki > 100000 nM T77365 CLT4W1 723688 Ki = 160 nM T77365 CF91NC 740769 Ki = 3.09 nM T77365 CZN6S9 743974 EC50 > 31622.78 nM T77365 C34AJP 747275 Ki > 100000 nM T77365 CZ6R2E 747391 Ki = 13 nM T77365 COW21P 750351 Ki = 1470 nM T77365 CDQH14 767064 Ki > 100000 nM T77365 CFA26R 785306 Ki > 100000 nM T77365 C08SPY 814471 Ki = 1300 nM T77365 CJW1K9 828537 Ki = 130 nM T77365 CJDR47 847241 Ki = 300 nM T77365 C8Y4NV 851050 Ki = 19000 nM T77365 CC94MT 851051 Ki = 1530 nM T77365 CCM2J1 851052 Ki = 610 nM T77365 CNJC61 853426 Ki = 43 nM T77365 CC1M8O 856282 Ki = 160 nM T77365 CE16YW 856297 Ki = 151 nM T77365 C50HPR 856323 Ki = 267 nM T77365 C2TDG1 883547 Ki = 350 nM T77365 CHJV30 906099 Ki > 1000 nM T77365 C2GDI3 912914 Ki = 31.62 nM T77365 C1WHL8 916396 Ki = 89 nM T77365 C7YQ1A 917384 Ki = 87 nM T77365 C5QFM2 933735 Ki = 39.81 nM T77365 CRSL39 1025219 Ki > 100000 nM T77365 CPV53L 1082196 Ki = 100 nM T77365 C56YAK 1084663 Ki > 100000 nM T77365 CWPQ69 1086298 Ki = 2700 nM T77365 C4H9ET 1160309 Ki = 1584.89 nM T77365 CCT83A 1259943 Ki > 100000 nM T77365 C2XHK6 1264044 Ki = 32 nM T77365 CV79ER 1350383 Ki = 38018.94 nM T77365 CC70IB 1482927 Ki = 2511.89 nM T77365 C5P2TF 1487654 Ki > 10000 nM T77365 CI5J9A 1487656 Ki > 10000 nM T77365 CH70DU 1504749 Ki = 150 nM T77365 C4M8RY 1505193 Ki = 31 nM T77365 C8RV0X 1505221 Ki = 49 nM T77365 CM80QJ 1509337 Ki = 19 nM T77365 CO7S1B 1532293 Ki = 740 nM T77365 CF4MA7 1598462 Ki = 1000 nM T77365 CC59EU 1635730 Ki = 14000 nM T77365 C5D6HZ 1722573 Ki > 100000 nM T77365 C3MYI6 1780327 Ki = 15.14 nM T77365 CZA28U 1856915 Ki = 300 nM T77365 CT9Q1W 1857272 Ki = 17000 nM T77365 CO1FZ7 2079368 Ki > 100000 nM T77365 CMW1F0 2302856 Ki = 2700 nM T77365 CK8T0W 2748282 Ki > 10000 nM T77365 CC8G6P 2778810 Ki = 54300 nM T77365 C1AFP2 2789377 Ki = 5011.87 nM T77365 CD84EF 2817023 Ki = 12 nM T77365 C5NV8W 2847378 Ki > 100000 nM T77365 C58MIA 2857005 Ki = 560 nM T77365 C51GNW 2874872 Ki > 10000 nM T77365 CHWU72 2910343 Ki > 100000 nM T77365 C3XOB4 2917156 Ki = 60 nM T77365 CRQD46 2942088 Ki = 15000 nM T77365 CFX98T 2947810 Ki = 400 nM T77365 CSB2Z3 2967583 Ki = 630.96 nM T77365 CW2KB4 2982214 Ki = 630 nM T77365 CYX74K 2985155 Ki = 2200 nM T77365 C40JOV 2986621 Ki = 41000 nM T77365 CS6Q9H 2989397 Ki > 100000 nM T77365 CRO73B 2989630 Ki = 1180 nM T77365 C9UYC2 3000506 Ki = 124 nM T77365 C80EBV 3000516 Ki = 2534 nM T77365 C5XTM7 3013233 Ki = 900 nM T77365 C5TCF2 3044933 Ki = 210 nM T77365 CBM9N7 3071852 Ki = 18 nM T77365 CPNR09 3162488 Ki = 2890 nM T77365 C4ZI9K 3162667 Ki > 1000 nM T77365 CQ0KB2 3240564 Ki = 1000 nM T77365 CSVD14 3349998 Ki = 130 nM T77365 C8LGP4 3462291 Ki = 5011.87 nM T77365 CI30FE 3463042 Ki = 59 nM T77365 CG8RD0 3636010 EC50 = 13800 nM T77365 CSR1K4 3751417 Ki = 403 nM T77365 CGRK30 3829487 Ki = 4677.35 nM T77365 CLYH52 4358247 Ki = 1258.93 nM T77365 CUE3C9 4382765 Ki = 287 nM T77365 CF7I6D 4388935 Ki = 120000 nM T77365 CWP4O1 4412077 Ki = 287 nM T77365 CKH03U 4480217 Ki = 210 nM T77365 C4W0UE 4610952 Ki > 100000 nM T77365 CUM2W1 4613432 Ki = 890 nM T77365 CE0OD3 4652320 Ki = 190 nM T77365 C3M4OS 4780194 Ki > 100000 nM T77365 CE38NO 4839305 Ki = 2951.21 nM T77365 CPW02K 4885273 Ki = 200 nM T77365 CGJ2D4 4897865 Ki = 1230.27 nM T77365 CD31SF 4976464 Ki > 100000 nM T77365 C70ILQ 5033052 Ki = 348 nM T77365 CV4M8K 5244097 Ki > 10000 nM T77365 CR3IW1 5296699 Ki = 17000 nM T77365 CZB37F 5311431 Ki > 10000 nM T77365 C25LIE 5373676 Ki = 1800 nM T77365 C2T6UE 5373687 Ki > 10000 nM T77365 CFL28J 5389037 Ki = 1584.89 nM T77365 CD1Y0R 5392003 Ki = 79.43 nM T77365 CY6T1I 5399631 Ki = 50.12 nM T77365 CPZ4C5 5399634 Ki = 7943.28 nM T77365 CU6WG0 5413075 Ki = 25.12 nM T77365 CT9QS8 5416642 Ki = 31.62 nM T77365 CV78YJ 5425546 Ki = 1995.26 nM T77365 C0A9NF 5462118 Ki = 54 nM T77365 CF7C6E 5462119 Ki = 1 nM T77365 C80UKF 5467768 Ki = 460 nM T77365 CX43YD 5468910 Ki = 440 nM T77365 C6F4HO 5571121 Ki = 19.95 nM T77365 CATJ51 5727370 Ki = 3981.07 nM T77365 CC0P2D 6032251 Ki = 316.23 nM T77365 CKN8G1 6402968 Ki = 3981.07 nM T77365 CTK1P2 6439089 Ki = 190 nM T77365 C6NP7A 6484523 Ki = 1200 nM T77365 CPM72Y 6621324 Ki = 2511.89 nM T77365 CNE6A5 6918429 Ki = 56 nM T77365 CD2XL9 7082904 Ki = 44000 nM T77365 CU6KF1 7162129 Ki > 100000 nM T77365 C82RXW 8024293 Ki = 36000 nM T77365 C70MOW 9246778 Ki = 3500 nM T77365 C3O8GK 9247074 Ki = 3600 nM T77365 CV6MD7 9268497 Ki = 25000 nM T77365 C32LEZ 9497523 Ki = 1.4 nM T77365 CRH9D2 9586623 Ki = 5011.87 nM T77365 CTYZ64 9798764 Ki = 670 nM T77365 CKNT38 9801343 Ki = 1390 nM T77365 C0BJD9 9803226 Ki = 190 nM T77365 CRHL94 9803956 Ki > 5000 nM T77365 C2EJD7 9803992 Ki = 594 nM T77365 C92LUT 9805713 Ki = 860 nM T77365 CQ51AF 9808834 Ki = 20.1 nM T77365 C98ERU 9814428 Ki = 3.3 nM T77365 CM96GZ 9814538 Ki = 6.6 nM T77365 CZR3N8 9816781 Ki = 52 nM T77365 CF8V3M 9818556 Ki = 2 nM T77365 C0JI5S 9819926 Ki = 5011.87 nM T77365 CVLM89 9821879 Ki = 290 nM T77365 C0TS3U 9822488 Ki = 690 nM T77365 C2O9IQ 9822747 Ki = 1195 nM T77365 C6O8QC 9823491 Ki = 3 nM T77365 C09BDM 9823602 Ki = 490 nM T77365 CAQS87 9824812 Ki = 545 nM T77365 CK0FX6 9825550 Ki = 2.239 nM T77365 CO51GB 9827315 Ki = 93.33 nM T77365 CUG62V 9827467 Ki = 39 nM T77365 CFLM79 9834242 Ki = 194 nM T77365 CLMN73 9834888 Ki = 12 nM T77365 CTGU01 9835359 Ki = 18 nM T77365 C9BZC8 9836304 Ki = 239 nM T77365 CS6IN9 9839378 Ki = 230 nM T77365 CFXZ58 9839545 Ki = 1.11 nM T77365 C4TOH3 9841364 Ki = 9.8 nM T77365 C25KVI 9842054 Ki = 16 nM T77365 C12UDF 9843101 Ki > 10000 nM T77365 CKZ07C 9843424 Ki > 100000 nM T77365 CU6Q8E 9844060 Ki = 912 nM T77365 CDO4W1 9844103 Ki = 2140 nM T77365 CUYI26 9844693 Ki = 3330 nM T77365 CZDJ43 9845174 Ki = 1.5 nM T77365 CRLO45 9850648 Ki = 784 nM T77365 C2F8KA 9850900 Ki = 642 nM T77365 CG63AF 9851062 IC50 = 100 nM T77365 C26KJD 9851372 IC50 = 28 nM T77365 C3MDK9 9856035 Ki = 70.4 nM T77365 CKEA76 9856296 Ki = 108 nM T77365 CUB8T7 9857266 Ki = 12 nM T77365 CUZL86 9857422 Ki = 1.9 nM T77365 CP50JH 9857698 Ki = 3 nM T77365 CUO04X 9857735 Ki = 2 nM T77365 CVR73U 9857814 Ki = 5 nM T77365 C1KP5W 9858219 Ki = 6.8 nM T77365 C52DIU 9858247 Ki = 12 nM T77365 CYXI30 9858577 Ki = 31 nM T77365 C6IK1X 9858578 Ki = 8.5 nM T77365 CUGV50 9860013 Ki = 1.4 nM T77365 CZRS26 9863617 Ki = 20 nM T77365 CZH74F 9864445 Ki = 1350 nM T77365 CTK0Z8 9865923 Ki > 6000 nM T77365 CBZA46 9865924 Ki = 380 nM T77365 CX04UV 9865974 Ki = 1280 nM T77365 CZN45Y 9865975 Ki = 56.8 nM T77365 CV19SJ 9868763 Ki = 1025 nM T77365 CRJ04W 9868991 Ki = 110 nM T77365 C7ARK4 9870396 Ki = 1400 nM T77365 CT8EK5 9870616 Ki = 710 nM T77365 CQR53Y 9870718 Ki = 431 nM T77365 CG47TN 9870719 Ki = 58.9 nM T77365 C3JW1Y 9873482 Ki = 0.05 nM T77365 C36IFS 9879687 Ki = 4 nM T77365 CTJ2A0 9879745 Ki = 27 nM T77365 C1ZH7A 9880379 Ki = 8 nM T77365 CQ0T4V 9880392 Ki = 8.2 nM T77365 CYPJ74 9880921 Ki = 6.6 nM T77365 C5URA3 9881967 Ki > 10000 nM T77365 CB26YS 9883190 Ki = 360 nM T77365 CL6AW0 9886589 Ki = 1070 nM T77365 CS0DL9 9887467 Ki = 440 nM T77365 CZN50C 9887859 Ki = 60 nM T77365 CLIE16 9890003 Ki = 796 nM T77365 C7C5VN 9890439 Ki = 400 nM T77365 C8LSD7 9893136 Ki = 1600 nM T77365 C36BVX 9895687 IC50 = 9 nM T77365 CE5G7X 9900111 Ki = 19 nM T77365 CF6M1U 9900245 Ki = 5.7 nM T77365 C7AE0U 9901099 Ki = 3 nM T77365 CCI2A0 9901100 Ki = 6 nM T77365 C0RCP7 9901171 Ki = 2.5 nM T77365 CDPV97 9901196 Ki = 4 nM T77365 CW8PY4 9901260 Ki = 2.7 nM T77365 C48DTC 9901296 Ki = 76 nM T77365 CJKD76 9901497 Ki = 3.9 nM T77365 CW8Z9K 9901700 Ki = 1.8 nM T77365 CMKV90 9901760 Ki = 23 nM T77365 CTU57Q 9902350 IC50 > 10000 nM T77365 CA52RY 9902562 Ki = 8.5 nM T77365 CJ3OC1 9902563 Ki = 2.2 nM T77365 CE4G3C 9903342 Ki = 23 nM T77365 C7YM0O 9904456 Ki = 1.2 nM T77365 CF54HI 9904688 Ki = 16 nM T77365 CR4SN0 9910158 Ki = 180 nM T77365 CDN1R5 9910926 Ki = 1220 nM T77365 CDM8F9 9911298 Ki = 1120 nM T77365 C37VQP 9911385 Ki = 7880 nM T77365 C3W0YI 9912318 Ki = 0.6 nM T77365 CC9FE0 9912816 Ki = 19.95 nM T77365 CUM73L 9921668 Ki = 3.1 nM T77365 CMGL57 9923269 Ki = 1.7 nM T77365 CO7FP5 9924271 Ki = 4160 nM T77365 C8CU7X 9924272 Ki = 2020 nM T77365 CO52VW 9924325 Ki = 3580 nM T77365 CLK76N 9924994 Ki > 10000 nM T77365 CA4OK7 9925574 Ki = 1.3 nM T77365 CXWU86 9929340 Ki = 676 nM T77365 CDQN01 9929405 Ki = 799 nM T77365 C7X1TD 9929470 Ki = 381 nM T77365 C1R8JD 9930130 Ki = 22 nM T77365 C8TMY5 9932840 Ki = 3.1 nM T77365 CE1B3K 9934039 Ki = 980 nM T77365 CJ5YV8 9935943 Ki = 39 nM T77365 CO3MX7 9935978 Ki = 95.2 nM T77365 CY82JD 9936058 Ki = 1970 nM T77365 CR05XW 9936467 Ki = 3100 nM T77365 CL73VJ 9944058 Ki = 57 nM T77365 CJCR41 9944894 Ki = 4 nM T77365 COH51K 9945155 Ki = 57 nM T77365 CW4NR7 9945226 Ki = 2.3 nM T77365 CD4SZ1 9945283 Ki = 150 nM T77365 CABF84 9945542 Ki = 10 nM T77365 CL3MY6 9946338 Ki = 7220 nM T77365 CBZG96 9949541 Ki = 1 nM T77365 C1VU2P 9949650 Ki = 754 nM T77365 C4MSO1 9950776 Ki = 550 nM T77365 C9F7BL 9953799 Ki = 1040 nM T77365 C2KD6M 9954747 Ki = 16.1 nM T77365 C8WR2V 9955052 Ki = 143 nM T77365 C24IWK 9955121 Ki = 1.9 nM T77365 C7GH6I 9957239 Ki = 1518 nM T77365 CE0N2P 9965093 Ki = 2.1 nM T77365 CGK3L2 9965998 Ki = 11 nM T77365 CE3O1U 9966890 Ki = 7 nM T77365 CND8Q6 9967146 Ki = 2 nM T77365 CO1NR5 9967147 Ki = 3 nM T77365 CPGT28 9967620 Ki = 3.7 nM T77365 C2UF7H 9968253 Ki = 4.1 nM T77365 CNQ6C7 9969880 Ki = 6 nM T77365 CE9X8F 9969881 Ki = 3 nM T77365 CMZ6X7 9970667 Ki > 10000 nM T77365 CNE43U 9970832 Ki = 0.6 nM T77365 CVR5X8 9974009 Ki = 161 nM T77365 CZE6O5 9975036 Ki = 21 nM T77365 CZVI16 9976651 EC50 = 15848931.92 nM T77365 C5SZL7 9978117 Ki = 29 nM T77365 CLI90J 9981945 Ki = 8270 nM T77365 C5F1IV 9985321 Ki > 1000 nM T77365 C06EVM 9995603 Ki = 646 nM T77365 CP0E1S 9996282 Ki = 3.6 nM T77365 CJ83TP 9999033 Ki > 100000 nM T77365 CMP5T0 10007115 Ki = 305 nM T77365 C2WSC5 10014953 Ki > 10000 nM T77365 CPAT84 10020580 Ki = 5.7 nM T77365 CM3OS9 10021401 EC50 = 30 nM T77365 CA4X5Z 10026670 Ki = 0.12 nM T77365 C9E4GW 10029879 Ki > 5000 nM T77365 C7SA9X 10037104 EC50 = 7600 nM T77365 C5PF2I 10038941 Ki = 0.1 nM T77365 CP2ZS6 10039961 Ki > 10000 nM T77365 CJZY04 10040075 Ki = 6800 nM T77365 CX32QD 10046002 Ki = 1400 nM T77365 CLRM29 10046145 Ki = 5 nM T77365 CU7EA4 10047690 Ki = 91 nM T77365 C3X1QT 10050031 Ki = 0.19 nM T77365 C9SM7V 10052252 Ki > 5000 nM T77365 C1I2LX 10062252 Ki > 10000 nM T77365 CM39QU 10063481 Ki = 147 nM T77365 CJW0D6 10063525 Ki = 6530 nM T77365 C7EKU9 10063737 Ki > 10000 nM T77365 CGE17I 10065148 Ki = 2.1 nM T77365 C1W0YH 10083550 Ki = 4750 nM T77365 CQ7TL1 10084926 Ki = 49.5 nM T77365 CSF1K3 10085767 Ki = 1600 nM T77365 C1LKV6 10085895 Ki = 161 nM T77365 C5WKF0 10086435 Ki = 13000 nM T77365 C8AO2Y 10106813 Ki = 250000 nM T77365 C42KUZ 10108084 Ki = 5160 nM T77365 C4EMH7 10110033 Ki = 35 nM T77365 CTCI65 10110171 Ki = 44 nM T77365 CXDU75 10112838 Ki = 16 nM T77365 CS2O8Q 10114735 Ki = 1.4 nM T77365 CT72WX 10117199 Ki = 40 nM T77365 CAZJ75 10118562 Ki = 12.6 nM T77365 CCT64M 10122714 IC50 = 11 nM T77365 CDK7G2 10126504 Ki = 14.7 nM T77365 CFI6P8 10126989 Ki = 38 nM T77365 CWV6U7 10127218 Ki = 3.2 nM T77365 C57JMI 10127905 Ki = 5.1 nM T77365 C78NYU 10131882 IC50 > 10000 nM T77365 C5WDR4 10132256 Ki = 2700 nM T77365 CIN47Q 10132473 Ki = 6 nM T77365 C5JC6Y 10132529 Ki = 8 nM T77365 CJ98UF 10134958 Ki = 6 nM T77365 CVKA84 10135831 Ki = 62 nM T77365 C5HN6X 10146937 IC50 = 5 nM T77365 C1AU0B 10150517 Ki > 5000 nM T77365 CTH9N8 10150788 Ki = 4.8 nM T77365 C2KY9X 10152242 Ki = 1.1 nM T77365 C9TEB2 10152925 Ki = 2.3 nM T77365 CZ17TE 10153190 Ki > 1000 nM T77365 C6IC0Y 10154604 Ki = 2570 nM T77365 CBY63V 10155413 Ki = 2.2 nM T77365 C7OC0T 10156654 IC50 > 10000 nM T77365 CK2BC6 10157187 Ki = 27 nM T77365 CB9W7J 10158069 Ki = 15 nM T77365 C7J5EN 10158974 Ki > 5000 nM T77365 CE5I2B 10159082 Ki = 2 nM T77365 CL9X0J 10161370 Ki = 4 nM T77365 CQY65K 10161974 Ki = 0.7 nM T77365 CRVU75 10164201 Ki > 5000 nM T77365 CO9K0X 10169297 IC50 = 5 nM T77365 CNGC14 10173234 Ki = 6 nM T77365 CQFV72 10174023 Ki = 5 nM T77365 CL4S8Q 10174142 Ki = 17.9 nM T77365 C4FNY6 10175278 Ki > 1000 nM T77365 C02RZC 10178449 Ki = 27 nM T77365 CWF7V8 10179603 Ki = 73 nM T77365 C4GOP3 10180118 IC50 > 10000 nM T77365 CJB32O 10181038 Ki = 1.6 nM T77365 CSZ2C7 10193594 Ki = 11.5 nM T77365 CVR7Y3 10195616 Ki = 1.6 nM T77365 C5NOP9 10196114 Ki > 200 nM T77365 CQ28MK 10198863 EC50 = 30 nM T77365 CRY0O1 10200261 EC50 = 23 nM T77365 C5C1RP 10200381 Ki = 4 nM T77365 CW1IU4 10202273 Ki = 12 nM T77365 CB19DN 10203891 Ki = 1 nM T77365 C84MZR 10204847 Ki = 223.87 nM T77365 CBR34L 10206584 Ki = 8 nM T77365 C21NHP 10212625 IC50 = 7 nM T77365 C0EXW6 10216181 Ki = 6.2 nM T77365 C6MYG7 10216962 Ki = 3.3 nM T77365 CN9W0F 10225178 Ki = 9.5 nM T77365 CJ8SG2 10225240 Ki = 50 nM T77365 C8R9BW 10233870 IC50 = 6 nM T77365 CQXC61 10234071 IC50 = 33 nM T77365 CXH8W0 10236339 Ki = 7 nM T77365 C6A8EB 10237267 Ki = 39 nM T77365 COJY26 10238586 Ki = 7.1 nM T77365 CSFU89 10243194 EC50 = 5900 nM T77365 CP7K3D 10246959 Ki = 0.31 nM T77365 C5RKX3 10247091 Ki > 100000 nM T77365 C2HVY5 10248379 Ki = 363 nM T77365 CH7VN4 10249674 Ki = 0.13 nM T77365 C0TXB5 10250190 Ki = 46600 nM T77365 C0CG8M 10253877 Ki = 2500 nM T77365 CGMN21 10254700 Ki = 20.4 nM T77365 CT41UJ 10256007 EC50 = 97 nM T77365 C9RSB2 10256116 Ki = 6200 nM T77365 CS80UL 10257979 Ki = 5128.61 nM T77365 CXE9U4 10264070 Ki = 58000 nM T77365 C86SHK 10264202 Ki = 490 nM T77365 CRL70U 10266501 Ki = 170 nM T77365 CF1UN5 10267860 Ki = 73 nM T77365 CA3S5M 10269139 IC50 > 10000 nM T77365 CN40IZ 10269215 Ki = 1 nM T77365 CWQ12V 10269216 Ki = 1 nM T77365 CYCI04 10269418 Ki = 1 nM T77365 CA1U9H 10269806 Ki = 6 nM T77365 C2CQK6 10270416 Ki = 1 nM T77365 CMH98A 10270860 Ki = 9 nM T77365 C2YD7R 10277683 Ki = 1.1 nM T77365 C3MG6S 10278807 Ki = 0.9 nM T77365 CG45IP 10287757 Ki = 2 nM T77365 CVND46 10287779 Ki = 2 nM T77365 C6W1SH 10287801 Ki = 5.4 nM T77365 CEX96C 10288019 Ki = 2.5 nM T77365 CLOQ10 10288204 Ki = 1.9 nM T77365 C0HIU5 10288740 Ki = 1.9 nM T77365 C6ATR8 10288990 Ki = 2 nM T77365 CIQ18W 10291002 Ki = 1 nM T77365 CI5LZ3 10291235 Ki = 349 nM T77365 C8ZVR9 10291405 Ki = 2 nM T77365 C0VY4L 10291948 Ki = 1670 nM T77365 C8RM9P 10292899 EC50 = 0.001 nM T77365 CD90SM 10294620 Ki = 2 nM T77365 C40WZO 10296638 Ki = 9.4 nM T77365 CZ58YA 10297926 Ki = 76 nM T77365 CXGB86 10301670 Ki = 0.4 nM T77365 CT1Q8X 10305241 IC50 = 17 nM T77365 C6PDF4 10305890 IC50 = 0.4 nM T77365 CI2E8K 10308937 Ki > 5000 nM T77365 C8US4I 10310635 Ki = 0.7 nM T77365 C8BO9X 10310768 Ki > 5000 nM T77365 CE2Q0P 10310914 Ki = 3.1 nM T77365 CBSE14 10311510 Ki = 23 nM T77365 C0H5MU 10316176 Ki = 196 nM T77365 CWN27R 10317753 Ki = 6.5 nM T77365 CXY40F 10318983 Ki = 0.18 nM T77365 CYM1D2 10330676 EC50 = 27500 nM T77365 CZ81IA 10342970 Ki = 3080 nM T77365 C0XHI4 10345159 Ki = 5660 nM T77365 C5Y1NM 10345700 Ki = 6.5 nM T77365 C7IPE9 10346511 Ki = 200 nM T77365 CF4UB5 10357057 Ki = 20 nM T77365 CD7C2A 10359522 Ki = 119 nM T77365 C8U2HR 10361312 Ki = 28900 nM T77365 C1RFV6 10362099 Ki = 1.5 nM T77365 C2R9YK 10369458 Ki = 29800 nM T77365 CCQ79O 10376254 EC50 = 8300 nM T77365 C63XFI 10377425 EC50 = 5000 nM T77365 CHZ32J 10377463 Ki = 11.22 nM T77365 CYK1L7 10378132 EC50 = 1400 nM T77365 CV4UJ5 10381286 Ki = 22900 nM T77365 C5HPZ3 10387088 Ki = 2540 nM T77365 C73CUW 10387599 EC50 = 12900 nM T77365 CUP34N 10388920 Ki = 49.9 nM T77365 CR53SP 10390495 Ki = 6.4 nM T77365 C7LG8M 10400587 EC50 = 3100 nM T77365 C5F4WP 10403711 EC50 = 22.9 nM T77365 CEU64Y 10425294 Ki = 46000 nM T77365 CAJ68I 10426659 Ki = 3150 nM T77365 CWUB34 10431614 Ki = 180 nM T77365 C9D5ZQ 10431643 EC50 = 7500 nM T77365 CO4H0C 10436433 EC50 = 1.4 nM T77365 CVE4Z0 10444746 Ki = 292000 nM T77365 CP4XJ5 10445452 Ki = 0.1 nM T77365 CI2HT6 10447827 Ki = 10000 nM T77365 CX0E9Q 10448644 Ki = 21700 nM T77365 CSD86M 10449535 EC50 = 26.8 nM T77365 C8XFL5 10449783 Ki > 10000 nM T77365 CK9FA7 10453097 Ki = 120 nM T77365 CM4C2X 10455080 Ki = 64 nM T77365 CGM46Y 10455852 Ki = 43 nM T77365 CI9UO8 10467925 Ki = 8400 nM T77365 CI3LE9 10471721 Ki = 849 nM T77365 C5Y6IP 10472803 Ki = 242 nM T77365 CBGS14 10492556 Ki = 1600 nM T77365 C93CAI 10494738 Ki > 10000 nM T77365 CHC23X 10505816 Ki = 101 nM T77365 CT4E5Q 10518459 Ki = 2400 nM T77365 C9OJF7 10522801 Ki = 5051 nM T77365 C08OQV 10528161 IC50 = 300 nM T77365 CCP12B 10537885 Ki > 10000 nM T77365 CJ8H1E 10538858 Ki = 40 nM T77365 CFOS68 10539663 Ki = 2608 nM T77365 CQIC13 10539682 Ki > 10000 nM T77365 C5ATC3 10541585 Ki = 14.6 nM T77365 CA2BP3 10544916 Ki = 11 nM T77365 CA8P6H 10547577 Ki = 4140 nM T77365 C53QCT 10554064 Ki = 1260 nM T77365 C2K6RI 10562783 Ki = 230 nM T77365 C37VFQ 10565553 Ki = 18.7 nM T77365 C3C8WE 10565773 Ki = 5750 nM T77365 CC84VI 10567830 Ki = 218 nM T77365 CZ7W5I 10569328 Ki = 1200 nM T77365 CVW26Q 10570266 Ki = 11400 nM T77365 C2T8YC 10572535 IC50 = 60 nM T77365 CL23DC 10580789 Ki = 2030 nM T77365 CEW4T3 10587109 Ki = 2.8 nM T77365 C02GZY 10601859 Ki = 200 nM T77365 CS2VT6 10605011 Ki = 3600 nM T77365 CSO52M 10613752 Ki = 11200 nM T77365 C6M1NH 10613770 Ki = 72 nM T77365 C2N5UX 10616023 Ki = 9.1 nM T77365 CL8WG1 10617844 Ki = 5400 nM T77365 CJ06HI 10618828 Ki = 15 nM T77365 CGMH35 10619822 Ki = 88.2 nM T77365 C3AUH2 10620944 Ki = 7440 nM T77365 C8JB3I 10623248 Ki = 80 nM T77365 CY6QP1 10626463 Ki > 10000 nM T77365 C7QWO6 10637742 Ki = 1.6 nM T77365 C78YHS 10641040 Ki = 156 nM T77365 CP86LA 10641062 Ki = 329 nM T77365 C7LN3U 10642208 Ki = 1370 nM T77365 CL03QM 10643254 Ki > 10000 nM T77365 C8O4LD 10645750 Ki = 2.7 nM T77365 C8O2UT 10647227 Ki = 95 nM T77365 CBI7X5 10659581 Ki = 1.9 nM T77365 C8NCG3 10661707 Ki = 45 nM T77365 CKG51X 10663067 Ki = 1900 nM T77365 C0U2LA 10665761 Ki = 13 nM T77365 CHQ6B9 10668865 Ki = 3.3 nM T77365 CGU6W0 10687707 Ki = 3277 nM T77365 C6SV1Y 10689930 IC50 = 14 nM T77365 CWJ60V 10691124 Ki = 19 nM T77365 C9B1PF 10696675 Ki = 105 nM T77365 CLZ7M1 10706862 Ki = 1500 nM T77365 C5EM0D 10709852 Ki = 376 nM T77365 C4PXZ8 10712345 IC50 = 3876 nM T77365 C07JSG 10720065 Ki = 187 nM T77365 CKIR94 10728732 Ki = 170 nM T77365 CJ8Z2O 10729354 Ki > 10000 nM T77365 CKMJ53 10732242 Ki = 1060 nM T77365 C7NXS3 10737168 Ki = 0.16 nM T77365 CB0L1T 10745111 Ki = 3260 nM T77365 C03CBY 10755990 Ki = 85.8 nM T77365 CSZW84 10757861 Ki = 490 nM T77365 CG67NI 10759742 Ki = 3800 nM T77365 CVM5F2 10760994 Ki = 5750 nM T77365 CWK2M9 10761106 Ki = 180 nM T77365 CUG21I 10761800 Ki = 13 nM T77365 CCZ4U8 10765059 Ki = 176 nM T77365 CO4XR0 10766011 IC50 = 90 nM T77365 CK0C8P 10767043 Ki = 16.6 nM T77365 C0FVU4 10767601 Ki = 470 nM T77365 C5B6KP 10769581 Ki = 348 nM T77365 CB9I0J 10778032 Ki > 10000 nM T77365 CIRS48 10778887 Ki = 49 nM T77365 C3GJ5Z 10779327 Ki = 2.51 nM T77365 CNC32V 10785815 Ki = 66 nM T77365 C79MNZ 10791347 Ki = 120 nM T77365 CYG2J5 10792296 Ki = 238 nM T77365 C7U4RN 10801510 Ki = 7000 nM T77365 C1AQO4 10801841 Ki = 1023 nM T77365 C3SCU6 10802472 Ki = 22500 nM T77365 C2N5AB 10812872 IC50 = 500 nM T77365 C7BT0O 10824674 Ki = 33 nM T77365 CQ01KP 10824688 Ki = 6500 nM T77365 C1TP5N 10828916 Ki > 10000 nM T77365 C7XJ0O 10831497 IC50 = 149 nM T77365 C6UP5K 10834513 Ki = 896 nM T77365 C2E6PX 10839228 Ki = 223 nM T77365 C20WTU 10839296 Ki = 70 nM T77365 C89OKC 10840167 Ki = 1640 nM T77365 C6GIK9 10847356 Ki = 210 nM T77365 C56NAP 10849482 Ki = 5000 nM T77365 C6CSZ4 10852375 Ki = 0.8 nM T77365 CE04SL 10852506 Ki = 0.78 nM T77365 C3I2WZ 10859484 Ki = 10 nM T77365 C3QWZ1 10862463 Ki = 1100 nM T77365 CZ7WJ9 10863425 Ki = 352 nM T77365 C4J8CR 10868826 Ki = 12100 nM T77365 C4HO6X 10874051 Ki = 3.1 nM T77365 C2B1MG 10878835 Ki = 682 nM T77365 C1AL7H 10884000 Ki = 22 nM T77365 CCV1Q4 10884004 EC50 = 800 nM T77365 CN8J0Y 10884265 Ki = 680 nM T77365 CY62BK 10884803 Ki = 1115 nM T77365 CP0M3N 10892251 Ki > 10000 nM T77365 CLGC13 10893465 Ki > 10000 nM T77365 CIG9Z2 10895416 Ki = 140 nM T77365 C2P1QB 10895565 Ki = 38 nM T77365 C2LV6K 10904370 Ki > 1000 nM T77365 CU93CT 10904839 Ki = 0.22 nM T77365 C3KOX6 10905184 Ki = 110 nM T77365 CKV30L 10905799 Ki = 148 nM T77365 CH52LS 10906943 Ki = 42 nM T77365 C4H8PS 10914466 Ki > 10000 nM T77365 CI87AW 10915653 Ki = 180 nM T77365 CJ52TM 10916451 Ki = 4.63 nM T77365 CS58FH 10917575 Ki = 4.1 nM T77365 CVFL61 10918042 Ki = 66 nM T77365 CGXE04 10925715 Ki = 2600 nM T77365 CQXA29 10926253 Ki = 135 nM T77365 CJB64E 10927693 Ki = 200 nM T77365 CFZ49H 10928011 Ki = 1.31 nM T77365 C1B6XL 10928182 Ki = 100 nM T77365 CG2N7W 10928649 Ki = 503 nM T77365 C7F8YE 10937272 Ki > 10000 nM T77365 C58CRE 10938276 Ki = 30 nM T77365 CG24MW 10938325 Ki = 1 nM T77365 C6FQ3L 10938608 Ki = 12 nM T77365 C8BLN4 10939224 Ki = 667 nM T77365 C5ORG7 10949999 Ki = 2140 nM T77365 CSE18R 10958838 Ki > 10000 nM T77365 CXWV50 10959335 Ki = 55 nM T77365 CY2OS9 10961304 Ki = 21 nM T77365 C7YVC5 10962009 Ki = 120 nM T77365 CAM58P 10968439 Ki > 10000 nM T77365 CLK8M1 10970782 Ki = 5610 nM T77365 CKE84F 10970819 Ki = 267 nM T77365 C7TUS2 10970979 Ki = 25800 nM T77365 CD16UB 10971099 Ki = 335 nM T77365 C9WLT0 10971427 Ki = 4.8 nM T77365 C6OFK0 10971806 Ki = 140 nM T77365 C4ZU8F 10971841 Ki = 42 nM T77365 CBW9J6 10972594 Ki = 4.4 nM T77365 C8F9LD 10979983 Ki > 10000 nM T77365 C4G0YQ 10982985 Ki = 121 nM T77365 C83XMH 10993869 Ki = 140 nM T77365 C6BH4T 10993916 Ki = 140 nM T77365 C9NP1R 10994142 Ki > 1000 nM T77365 C3F4TJ 10994183 Ki = 376 nM T77365 CSO19C 10994216 Ki = 43.9 nM T77365 C31HJV 10994317 Ki = 34 nM T77365 CH6Y5I 11000858 Ki = 4100 nM T77365 CMDB43 11004373 Ki = 150 nM T77365 CEP35L 11004986 Ki > 1000 nM T77365 CLR4B8 11005067 Ki = 1.1 nM T77365 C0KDE3 11014188 Ki = 423 nM T77365 C47IDH 11014608 Ki = 196 nM T77365 C46AKC 11014956 Ki = 3 nM T77365 C6EQD3 11015003 Ki = 60 nM T77365 C5BQ0H 11015572 Ki = 10.2 nM T77365 C30WTZ 11017082 Ki = 0.59 nM T77365 CI3E7D 11019436 Ki > 100000 nM T77365 C9TPE8 11022827 Ki = 720 nM T77365 C20KVX 11025671 EC50 = 5000 nM T77365 C8UPZ3 11026001 Ki = 163 nM T77365 CF5B8Z 11026358 Ki > 1000 nM T77365 CPD61T 11026434 Ki = 614 nM T77365 C12YXH 11027282 Ki = 75 nM T77365 CX28EA 11027412 Ki = 45 nM T77365 CPV27K 11027743 Ki = 29800 nM T77365 CW05DS 11028588 Ki > 1000 nM T77365 CHEA89 11037671 Ki = 0.43 nM T77365 CR7FM2 11037739 Ki = 111 nM T77365 CM9FK6 11037972 Ki = 40 nM T77365 CPB50W 11045730 Ki = 3200 nM T77365 C85NWI 11047444 EC50 = 500 nM T77365 CS8P0U 11048163 Ki = 100 nM T77365 CL1RP8 11048438 Ki = 324 nM T77365 CW7Q6U 11053743 Ki = 212 nM T77365 CL29NE 11056301 Ki = 584 nM T77365 CTZM01 11058084 Ki = 2500 nM T77365 CCS8A6 11058550 Ki = 180 nM T77365 CYZ83I 11059351 Ki = 91 nM T77365 CA91IB 11060260 Ki = 3.8 nM T77365 CM7TR4 11068963 Ki = 8530 nM T77365 C9KRQ1 11070905 Ki = 305 nM T77365 C7HIP2 11071159 Ki > 1000 nM T77365 CN5S7E 11078951 Ki > 1000 nM T77365 C1EJI0 11080491 Ki = 57 nM T77365 CKX4G6 11080788 Ki = 95 nM T77365 C4Y7NZ 11081189 Ki = 401 nM T77365 C83TJN 11090423 Ki = 385 nM T77365 CR3X1M 11091600 Ki = 15 nM T77365 C64PWO 11091632 Ki = 100 nM T77365 C15EQZ 11091783 Ki = 61 nM T77365 CZW34N 11099564 Ki = 96 nM T77365 CVDM13 11102838 Ki = 50 nM T77365 C0DXW3 11109201 Ki > 10000 nM T77365 CMY97P 11112381 Ki = 1560 nM T77365 C3Z5PU 11112543 Ki = 133 nM T77365 CJ21DZ 11112670 EC50 = 10400 nM T77365 C6RB5D 11112711 Ki = 1181 nM T77365 C3IFX4 11112849 Ki = 576 nM T77365 CR7X2T 11122708 Ki = 160 nM T77365 CLN23H 11123135 Ki > 1000 nM T77365 C06JLD 11123887 Ki = 352 nM T77365 C4CWA8 11133107 Ki > 1000 nM T77365 CJ86ZM 11133545 Ki = 695 nM T77365 CL19OW 11133804 Ki = 113 nM T77365 CTG5Y7 11133843 Ki = 50 nM T77365 C29UBQ 11143352 Ki = 489.78 nM T77365 CH4TG2 11144119 Ki > 1000 nM T77365 C9N1RL 11144868 Ki = 100 nM T77365 C72QCG 11145314 Ki = 50 nM T77365 C4AR0D 11150120 Ki > 10000 nM T77365 CVF8Z5 11151115 Ki > 10000 nM T77365 CH3LA7 11151693 Ki = 200 nM T77365 C79YSE 11153187 Ki > 1000 nM T77365 CM9SW5 11154129 Ki = 102 nM T77365 CLQR16 11157262 EC50 = 1.6 nM T77365 C1FVD5 11162618 Ki = 2.6 nM T77365 CNY65E 11163483 Ki = 9700 nM T77365 CJ0T6F 11163971 Ki = 22 nM T77365 C6ALI1 11164274 Ki = 1.1 nM T77365 CS0N2C 11164346 Ki = 214 nM T77365 CJN5M3 11168952 Ki = 2780 nM T77365 CPB62L 11174953 Ki = 28 nM T77365 C12UTW 11175566 Ki > 1000 nM T77365 CFL0O8 11177363 Ki = 51.8 nM T77365 CJ02LB 11178828 Ki = 4000 nM T77365 CHD65Q 11198201 Ki > 1000 nM T77365 CD7QP2 11199731 Ki = 20.6 nM T77365 C41PYH 11209919 Ki > 1000 nM T77365 C6JD3L 11210192 Ki > 10000 nM T77365 CL6EM0 11210971 Ki = 49.3 nM T77365 CV5Y6A 11214123 EC50 = 10.6 nM T77365 CUNM43 11220580 Ki = 2.8 nM T77365 C2D5RQ 11221675 Ki = 220 nM T77365 C3FP0D 11229946 Ki = 3.7 nM T77365 CK5P7G 11232232 Ki = 8.5 nM T77365 C3B4ZF 11232994 Ki = 2950 nM T77365 C9IHT1 11233411 Ki > 1000 nM T77365 CB6Y4A 11233413 Ki > 1000 nM T77365 C1KM3O 11244144 Ki = 13000 nM T77365 C57WSV 11244376 Ki = 179 nM T77365 CG0OL1 11254831 Ki = 3.6 nM T77365 CES2X9 11255221 Ki > 10000 nM T77365 CA4EP9 11255271 Ki > 10000 nM T77365 C7LS3R 11256992 Ki = 105 nM T77365 CCU71Z 11257069 Ki > 1000 nM T77365 C86XNQ 11260448 Ki = 1800 nM T77365 CH0U1C 11266371 Ki = 1400 nM T77365 CK7SM8 11266431 Ki > 10000 nM T77365 CL60TZ 11267343 Ki = 631 nM T77365 CDL7O5 11277831 Ki = 3800 nM T77365 CYWN16 11278445 Ki = 11 nM T77365 C45RAF 11289724 Ki > 10000 nM T77365 CGR1A8 11289861 Ki = 7 nM T77365 C48JAP 11290020 Ki = 228 nM T77365 C8B2RV 11290216 Ki = 1049 nM T77365 C5QDY9 11290412 Ki = 67 nM T77365 C8A0MT 11290634 Ki = 1725 nM T77365 CLW5H2 11301432 Ki > 10000 nM T77365 C3Y1OW 11302050 Ki = 28 nM T77365 CQ7O1I 11302588 Ki = 6100 nM T77365 CJS9C0 11304851 IC50 = 25000 nM T77365 C4PH8A 11306173 Ki = 3780 nM T77365 CJ4MT0 11311283 Ki = 110 nM T77365 CDC83I 11312454 Ki = 388 nM T77365 CX09ZQ 11312833 Ki > 10000 nM T77365 CGB03H 11313388 Ki = 47 nM T77365 C9KYQ4 11313397 Ki = 162 nM T77365 CCMS25 11313542 Ki = 120 nM T77365 CO1Q4Y 11313543 Ki = 19 nM T77365 CUS2N9 11313850 Ki > 1000 nM T77365 CX7QW0 11324734 Ki = 1200 nM T77365 C5UMJ9 11324754 Ki = 63 nM T77365 CMXN49 11328135 Ki = 1.5 nM T77365 CY8KX5 11329375 Ki = 1200 nM T77365 CGCJ09 11335341 Ki = 80 nM T77365 CJX89P 11348709 Ki > 1000 nM T77365 C1Q8NA 11348867 Ki = 208 nM T77365 C3TH4B 11352497 Ki = 5 nM T77365 CEI47X 11353406 Ki = 4000 nM T77365 C2Z8GE 11358739 Ki = 181 nM T77365 CRND96 11360082 Ki > 1000 nM T77365 CT8J7Q 11368737 Ki = 230 nM T77365 C8G3FO 11371101 Ki > 1000 nM T77365 CB8RU3 11380183 Ki = 0.6 nM T77365 C0M8KH 11380777 Ki > 10000 nM T77365 CB3J6T 11380878 Ki = 9.4 nM T77365 CRU3A7 11381738 Ki = 6.1 nM T77365 C3IHK7 11381773 Ki = 5 nM T77365 CR73JH 11382077 Ki = 9.2 nM T77365 CSD31L 11386134 Ki = 100 nM T77365 C8KD6J 11386951 EC50 = 3.1 nM T77365 C21UDI 11387030 Ki = 3200 nM T77365 CJ9WG8 11391873 Ki = 580 nM T77365 CK58UE 11391964 Ki = 14 nM T77365 CB2C4P 11392671 Ki = 2.2 nM T77365 CVAJ46 11393155 Ki = 3.5 nM T77365 CXPM05 11394389 Ki > 1000 nM T77365 C1CL4W 11404060 Ki = 1117 nM T77365 C6IVY0 11408692 Ki = 129 nM T77365 CLM04X 11412911 Ki > 10000 nM T77365 CD9PL7 11415171 Ki > 10000 nM T77365 C3NO7I 11415926 Ki = 1700 nM T77365 CS7ZX2 11416448 Ki = 1789 nM T77365 CCW60O 11420226 Ki = 781 nM T77365 CDVM74 11424338 Ki > 10000 nM T77365 C30ZXP 11426423 Ki = 4.3 nM T77365 CQ7H6Z 11427378 Ki > 10000 nM T77365 CPF8K7 11427490 Ki = 128 nM T77365 CPS9L6 11427880 Ki = 196 nM T77365 CF4H1A 11428535 Ki > 1000 nM T77365 C85LYP 11430418 IC50 > 1000 nM T77365 C1U0CT 11431149 Ki = 1955 nM T77365 CF8EN7 11437060 Ki = 210 nM T77365 CL7S1A 11439147 Ki = 1600 nM T77365 CZP97D 11440111 Ki = 0.8 nM T77365 C6CV1B 11452333 Ki > 1000 nM T77365 CA6YD2 11461202 Ki = 189 nM T77365 CZIN71 11462033 Ki = 196 nM T77365 C5M3SD 11463674 Ki > 1000 nM T77365 C5JTD0 11464552 Ki > 1000 nM T77365 C9CFK5 11465677 Ki > 1000 nM T77365 C9NP2C 11466670 Ki = 1700 nM T77365 CDY79C 11472819 Ki = 9.3 nM T77365 CK9VD0 11473488 Ki = 50 nM T77365 C9RK6X 11475577 Ki > 1000 nM T77365 C83XMS 11475769 Ki > 5000 nM T77365 C67UZW 11476550 Ki = 1 nM T77365 CE7JS1 11483771 Ki = 3.5 nM T77365 C2SY3I 11492651 Ki = 1520 nM T77365 CI4JC0 11492857 Ki = 303 nM T77365 CL49IS 11493754 Ki = 3500 nM T77365 CKN80I 11494063 Ki > 1000 nM T77365 C5FY2G 11494318 Ki = 51.6 nM T77365 CZ0FN7 11494993 Ki = 7503 nM T77365 CO32QT 11495161 Ki = 51 nM T77365 C1P7DN 11495410 Ki = 181.97 nM T77365 CH7UC9 11495611 Ki = 49 nM T77365 CJ8NX6 11495984 Ki = 213.8 nM T77365 CPIQ63 11497055 Ki = 38.9 nM T77365 C5LN1D 11497238 Ki = 42 nM T77365 C60KRJ 11498113 Ki = 52.48 nM T77365 C3YG6W 11500266 Ki = 3000 nM T77365 C6KL3S 11501678 Ki = 140 nM T77365 CD0T6O 11503200 Ki = 870 nM T77365 CQF31J 11503616 Ki = 131.83 nM T77365 C08TYB 11503979 Ki = 186.21 nM T77365 CL60QU 11505071 Ki = 79.43 nM T77365 C0WV8M 11507345 Ki > 10000 nM T77365 COG79X 11508049 Ki = 307 nM T77365 C5A8ZL 11508721 Ki = 776.25 nM T77365 C0AWD8 11508923 Ki = 231 nM T77365 C4DUQ1 11509299 Ki = 3715.35 nM T77365 CSLD98 11510702 Ki = 66.07 nM T77365 CO4B6S 11510891 Ki = 575.44 nM T77365 CLM6Q8 11511593 Ki = 31.62 nM T77365 C8GL1J 11511804 Ki > 1000 nM T77365 CH03ZF 11516748 Ki = 410 nM T77365 CD29AZ 11517013 Ki > 1000 nM T77365 C56UZA 11517635 Ki = 1023.29 nM T77365 C65MAZ 11519021 Ki = 2630.27 nM T77365 CMNY64 11519361 Ki = 263.03 nM T77365 C60VRX 11519405 Ki = 100 nM T77365 CT60SW 11522152 Ki = 3570 nM T77365 CS1M7B 11522670 Ki = 1790 nM T77365 CKIR86 11524078 Ki = 691.83 nM T77365 C4K0MX 11524240 Ki = 204.17 nM T77365 CQZ37L 11524264 Ki > 1000 nM T77365 CH9DU2 11524593 Ki = 890 nM T77365 C23LEU 11524637 Ki = 70 nM T77365 CIJA46 11524904 Ki = 43.65 nM T77365 C1CJ2S 11525283 Ki = 769 nM T77365 C3KE4L 11525368 Ki = 120.23 nM T77365 CYAW65 11525776 Ki = 275.42 nM T77365 CIH91Y 11525816 Ki = 323.59 nM T77365 CVR6D0 11527363 EC50 = 3 nM T77365 C21IUQ 11529194 Ki > 10000 nM T77365 CKC6F5 11529450 Ki = 379 nM T77365 CV2DP6 11530256 Ki = 5220 nM T77365 C46UMB 11531355 Ki = 4850 nM T77365 CG49ZV 11531449 Ki = 933.25 nM T77365 CEDZ81 11532717 Ki = 70 nM T77365 C6HAF9 11533237 Ki = 4300 nM T77365 C92FYA 11533614 IC50 = 2.7 nM T77365 C19JCF 11533636 Ki = 6570 nM T77365 CAZ51S 11533996 Ki = 107.15 nM T77365 CYWJ05 11535816 Ki > 10000 nM T77365 C8P2YI 11536894 Ki = 2400 nM T77365 C0Z9UA 11536947 Ki > 10000 nM T77365 CU38FS 11537425 Ki > 2500 nM T77365 CH43JG 11538373 Ki = 153 nM T77365 C5KDX9 11539152 Ki = 1870 nM T77365 CSY78B 11541413 Ki = 18.62 nM T77365 C16FKE 11544506 Ki > 2500 nM T77365 CT6C5U 11544894 Ki = 200 nM T77365 CW62MV 11545273 Ki = 125 nM T77365 C2QHP4 11545341 Ki = 560 nM T77365 CUD5B0 11546358 Ki = 810 nM T77365 C1U8RO 11547107 Ki = 150 nM T77365 C36DPX 11547533 Ki = 158.49 nM T77365 C5NOR2 11548192 Ki = 44.67 nM T77365 CB56MC 11548559 Ki = 19.95 nM T77365 CJ6QB9 11548714 Ki = 125.89 nM T77365 CPV7Y8 11553016 Ki > 10000 nM T77365 CO28UI 11553439 Ki = 1862.09 nM T77365 C3IET8 11553509 Ki = 47.86 nM T77365 C7OJ4E 11554182 Ki = 81.28 nM T77365 CHQ6F9 11554879 Ki = 627 nM T77365 C6CVK7 11555032 Ki > 1000 nM T77365 C2NVK8 11555329 Ki = 81.28 nM T77365 CF6E1O 11555462 Ki = 46.77 nM T77365 C5RHM0 11555968 Ki = 31.62 nM T77365 C7A9PY 11557440 Ki > 10000 nM T77365 C0VES1 11560202 Ki = 75 nM T77365 C7VD3G 11560510 Ki = 66 nM T77365 CIQK94 11560605 Ki = 3585 nM T77365 C5Q7TL 11561073 Ki = 169.82 nM T77365 CH3TK6 11561715 Ki = 120.23 nM T77365 CI9LM6 11561747 Ki = 489.78 nM T77365 CAN1B7 11562203 Ki = 53.7 nM T77365 C41AXZ 11565780 Ki = 365 nM T77365 CIR70L 11565927 Ki > 2500 nM T77365 CV9A8O 11566322 Ki = 1.4 nM T77365 C5JIZ0 11567699 Ki = 316.23 nM T77365 C93ANH 11568001 Ki = 64.57 nM T77365 C9WVP1 11568203 Ki = 450 nM T77365 C85MGW 11568359 Ki = 32.6 nM T77365 C9Y1JH 11568517 Ki = 891.25 nM T77365 CLV6H3 11568586 Ki = 1320 nM T77365 C37CAT 11569026 Ki = 8050 nM T77365 CQH34L 11569133 Ki = 56.23 nM T77365 CJM06D 11569877 Ki = 223.87 nM T77365 CVY43P 11570614 Ki = 158.49 nM T77365 CY3C0A 11573708 Ki = 33 nM T77365 C9VP0G 11574573 IC50 = 12 nM T77365 CZIP72 11574851 Ki = 1562 nM T77365 CQTN95 11575377 Ki = 7574 nM T77365 C7RA2X 11575498 Ki = 79 nM T77365 CAHB70 11576014 Ki = 26.3 nM T77365 CU3MW5 11576491 Ki = 104.71 nM T77365 CTW85Y 11576751 Ki = 489.78 nM T77365 CVQ19R 11577804 Ki = 292 nM T77365 CZ65AS 11580284 Ki = 110 nM T77365 C5JOW8 11580374 Ki = 527 nM T77365 C8Y9LA 11582537 Ki = 1100 nM T77365 CAR2U3 11582578 Ki = 140 nM T77365 C5I4RZ 11582697 Ki = 88 nM T77365 C8Q3FA 11583705 Ki = 89.13 nM T77365 CB8H3T 11584027 Ki = 107.15 nM T77365 C82YDZ 11584408 Ki = 707.95 nM T77365 C6D1MA 11584660 Ki > 3981.07 nM T77365 COVP09 11584826 Ki = 15.85 nM T77365 C0TFK3 11586663 Ki = 120 nM T77365 CM62BJ 11587409 Ki = 498 nM T77365 CYJ29E 11587927 Ki = 267 nM T77365 C8S2RC 11588630 Ki = 120 nM T77365 CN7T8C 11589094 Ki = 2770 nM T77365 CU0MX8 11589625 Ki = 60 nM T77365 CR6Y8H 11590025 Ki = 446.68 nM T77365 CH2TN6 11590097 Ki = 245.47 nM T77365 C5KX2E 11590453 Ki = 331.13 nM T77365 C9KJ2P 11590537 Ki = 20.42 nM T77365 CE2I5N 11591029 Ki = 32.36 nM T77365 CVE43I 11591558 Ki = 32.36 nM T77365 CI2ZO0 11591823 Ki = 89.13 nM T77365 CS1RK4 11595040 Ki = 2840 nM T77365 CNTA30 11595292 Ki = 77 nM T77365 CMF50J 11595592 Ki = 4073.8 nM T77365 C1ERP7 11595710 Ki = 1100 nM T77365 CGPE63 11596214 Ki = 5 nM T77365 CUXN24 11596614 Ki = 80 nM T77365 C31YOR 11596733 Ki = 180 nM T77365 C8OJ6R 11597583 Ki = 45 nM T77365 CVN1Y5 11601342 Ki > 10000 nM T77365 C1QJ4W 11602451 Ki = 1060 nM T77365 C80ZIV 11602914 Ki > 10000 nM T77365 C0A4FU 11604435 Ki = 186.21 nM T77365 CAC54T 11606834 Ki = 549 nM T77365 C21IGF 11608581 Ki = 83.7 nM T77365 CB06AO 11608818 Ki = 4930 nM T77365 C8LA0I 11609235 Ki = 6980 nM T77365 CPS1A9 11609536 Ki = 12 nM T77365 CWMD07 11610638 Ki = 290 nM T77365 CJW6N3 11610747 Ki = 11481.54 nM T77365 CC6GD1 11611016 Ki = 1000 nM T77365 CUIT18 11611298 Ki = 16.22 nM T77365 C6NID5 11611580 Ki = 460 nM T77365 CXB6L3 11611815 Ki = 1232 nM T77365 C42QLP 11611903 Ki > 10000 nM T77365 C0DGN8 11612118 Ki = 112.2 nM T77365 C2G4JX 11612320 Ki = 230 nM T77365 CC8Q7O 11612367 Ki = 1517 nM T77365 CE3ZL4 11613517 Ki = 85.11 nM T77365 CO5LH7 11617483 Ki = 83 nM T77365 CVW0B6 11618482 Ki = 1988 nM T77365 C39ZVR 11618633 Ki = 220 nM T77365 CF09KT 11619671 Ki = 4963 nM T77365 CLV26W 11623708 Ki = 334 nM T77365 C7AM8B 11623934 Ki = 634 nM T77365 CVL8P5 11625174 Ki = 4890 nM T77365 C2OD7U 11625772 Ki = 921 nM T77365 C35XDW 11625796 Ki = 60 nM T77365 C32ECV 11627336 Ki = 58.88 nM T77365 C2JW5N 11628044 Ki = 42.66 nM T77365 C02QTY 11630237 Ki > 10000 nM T77365 C0JOM4 11630922 Ki > 30000 nM T77365 C57HNQ 11631512 Ki = 48 nM T77365 CXSZ13 11632013 Ki = 94 nM T77365 CJ5OM1 11632785 Ki = 776.25 nM T77365 CJ02TL 11633189 Ki = 61 nM T77365 C7TFE5 11634270 Ki = 202 nM T77365 C2XD3T 11634901 Ki = 245.47 nM T77365 CX2B4O 11638430 Ki = 28 nM T77365 CFTH84 11638790 Ki > 2500 nM T77365 CH0K6M 11639132 Ki = 190 nM T77365 C42QLC 11639150 Ki > 10000 nM T77365 CXUQ86 11640487 Ki = 149 nM T77365 C80FAW 11640539 Ki = 45.71 nM T77365 CRB30J 11640595 Ki = 194.98 nM T77365 CG4J8D 11641051 Ki = 426.58 nM T77365 CM39TC 11641365 Ki = 1160 nM T77365 C85ZEB 11642035 Ki = 4897.79 nM T77365 CSG21Q 11645609 Ki = 4168.69 nM T77365 CQ6SY8 11646269 Ki = 1 nM T77365 CEC6Z2 11646441 Ki = 7671 nM T77365 C5BH2I 11647009 Ki = 1388 nM T77365 C9X5JF 11647607 Ki = 280 nM T77365 C0GX7S 11649117 Ki = 19.05 nM T77365 C3VZF7 11649145 Ki = 2630.27 nM T77365 CND50M 11649544 Ki = 30.9 nM T77365 CT6CW3 11650023 Ki = 326 nM T77365 CAX46N 11654460 Ki = 230 nM T77365 CIS7K1 11654461 Ki = 120 nM T77365 CC8X7R 11655061 Ki = 1300 nM T77365 CLU6I0 11656075 Ki = 25.7 nM T77365 CJ1X7N 11656185 Ki = 74.13 nM T77365 CFP83C 11656570 Ki = 89.13 nM T77365 CQ8SE2 11656950 Ki = 91.2 nM T77365 CM54YT 11657274 Ki = 2220 nM T77365 CWY7T6 11659363 Ki = 1830 nM T77365 C1JU7A 11659696 Ki > 2500 nM T77365 CPV35M 11660022 Ki = 367 nM T77365 C1JBL4 11660427 Ki = 1949.84 nM T77365 C1L0JI 11660995 Ki = 123.03 nM T77365 CU94XB 11662646 Ki = 429 nM T77365 CV39AR 11662965 IC50 = 62 nM T77365 C2BH0P 11663050 Ki = 67.61 nM T77365 C7D2CU 11663068 Ki = 15.49 nM T77365 CQ13SY 11663152 Ki = 3890 nM T77365 CGA72F 11663932 Ki > 10000 nM T77365 CC9YA7 11664137 Ki = 35.48 nM T77365 CI2SK9 11667107 Ki > 2500 nM T77365 CGI6Y3 11667703 Ki = 400 nM T77365 CB1Z8M 11667955 Ki = 57 nM T77365 C8SX1P 11667956 Ki = 25 nM T77365 CVPM67 11673316 Ki = 481.3 nM T77365 CX95RT 11674018 Ki = 120 nM T77365 CZ6V5H 11675684 Ki = 604 nM T77365 CU90TV 11675940 Ki = 325 nM T77365 CN04ER 11676113 Ki = 398.11 nM T77365 CAJ43T 11676986 Ki = 309.03 nM T77365 CL6A2N 11677252 Ki = 302 nM T77365 C24BUE 11677313 Ki = 12.02 nM T77365 CSTZ64 11677724 Ki = 39.81 nM T77365 CNH01O 11677816 Ki = 16.98 nM T77365 C16PMS 11678491 Ki > 10000 nM T77365 C7SJI1 11678808 Ki = 281.84 nM T77365 C1I6FC 11680901 Ki = 6330 nM T77365 CKU6E7 11681092 Ki = 450 nM T77365 CFD86C 11681113 Ki = 1020 nM T77365 CF54VW 11681354 Ki = 1700 nM T77365 CE8WD5 11681429 Ki = 1820 nM T77365 CI8AX3 11683024 Ki = 155 nM T77365 C94ZVJ 11683855 Ki = 45.71 nM T77365 CAS80N 11684443 Ki = 1230.27 nM T77365 CH30ES 11684672 Ki > 1000 nM T77365 C6UIK7 11684701 Ki = 26.92 nM T77365 CEU52V 11684979 Ki = 64 nM T77365 CI73GV 11685118 Ki = 48.98 nM T77365 C4SWY5 11687423 Ki > 10000 nM T77365 CYFJ70 11687483 Ki = 492 nM T77365 COX34C 11688036 Ki = 190 nM T77365 CT3JM9 11690561 Ki = 450 nM T77365 CI10PQ 11690712 Ki = 162 nM T77365 CFJ3X6 11690983 Ki = 95.5 nM T77365 CS9FL1 11693081 Ki = 426.58 nM T77365 CH6Q2D 11698898 Ki > 5000 nM T77365 CZ8I6J 11699025 Ki = 23.99 nM T77365 C2V3PS 11699353 Ki = 8 nM T77365 CWA0C8 11701717 Ki = 329 nM T77365 C69PJB 11702501 Ki = 4.7 nM T77365 C6HFY9 11703084 Ki = 200 nM T77365 CZ9IX2 11703893 Ki = 920 nM T77365 CZE9V5 11705261 Ki = 1100 nM T77365 C7BH9E 11705321 Ki = 1358 nM T77365 CDG61A 11706151 Ki = 60.26 nM T77365 CR6A2V 11709311 Ki = 1800 nM T77365 CX6E5A 11709650 Ki = 3080 nM T77365 C2LMK1 11711190 Ki = 570 nM T77365 CYI8O4 11711438 Ki > 1000 nM T77365 C72KXO 11711753 Ki = 1047.13 nM T77365 C80LHJ 11711754 Ki = 302 nM T77365 CPE2Q9 11713242 Ki = 40.74 nM T77365 C3RP8Y 11713561 Ki = 69.18 nM T77365 CIYJ64 11713673 Ki = 239.88 nM T77365 CY48OK 11715751 Ki > 10000 nM T77365 CUM0C9 11716303 Ki > 10000 nM T77365 CNR71Y 11717537 Ki = 350 nM T77365 CD72OJ 11717832 Ki > 1000 nM T77365 CCQ78R 11720113 Ki = 19.95 nM T77365 CDZ6P4 11720443 Ki = 724.44 nM T77365 CH5DB1 11720501 Ki = 282 nM T77365 CZR29N 11720513 Ki = 63.1 nM T77365 C5P4YO 11723628 Ki = 75.8 nM T77365 C3ZA9B 11728558 EC50 = 700 nM T77365 C9J4WY 11728711 Ki = 86 nM T77365 CAMT16 11728808 Ki = 40 nM T77365 CNT64M 11729275 Ki > 10000 nM T77365 CR80CF 11731871 Ki > 1000 nM T77365 C5GO4E 11732736 Ki = 24 nM T77365 CHW0A6 11733496 Ki = 60 nM T77365 CG7Y4O 11733556 Ki = 50 nM T77365 CF9Q7M 11733601 Ki = 31 nM T77365 CP2J9D 11738790 Ki = 4120 nM T77365 C43GFZ 11739282 Ki = 1.7 nM T77365 CEA40Z 11739584 Ki = 5.1 nM T77365 CCU3E4 11759055 Ki = 4300 nM T77365 CSR32T 11761221 Ki = 62 nM T77365 C7MD4U 11761823 Ki = 4 nM T77365 CGSN15 11762418 Ki = 249 nM T77365 CI82XE 11762982 Ki = 55 nM T77365 CB36OJ 11771503 Ki = 36 nM T77365 CE3D9A 11771825 Ki = 970 nM T77365 CT84IV 11774108 Ki > 1000 nM T77365 CO76RZ 11782906 Ki = 158 nM T77365 CLPT97 11784369 Ki = 306 nM T77365 CD68PT 11784529 Ki = 0.2 nM T77365 C7J6UF 11791862 Ki = 2210 nM T77365 CBZJ16 11798195 Ki = 65 nM T77365 CV7T3H 11798368 Ki = 115 nM T77365 C8ZRL4 11801496 Ki = 5140 nM T77365 C1ZQF6 11811544 Ki = 160 nM T77365 CCBY84 11811574 EC50 = 3600 nM T77365 CPMB38 11811761 Ki = 400 nM T77365 C82LEP 11812897 Ki = 495 nM T77365 C6ANG8 11813241 Ki = 0.12 nM T77365 CZ52VY 11813713 Ki = 223 nM T77365 CR46ZY 11821574 Ki > 10000 nM T77365 C20MGI 11823876 Ki > 10000 nM T77365 C4W2ID 11824950 Ki > 1000 nM T77365 C31FGJ 11826577 Ki = 53 nM T77365 C15NOJ 11826924 Ki = 40 nM T77365 CT3ZH4 11834222 Ki > 10000 nM T77365 CXLW54 11948707 Ki > 10000 nM T77365 C6Y3GI 11952504 Ki = 3605 nM T77365 C3Y9JS 11952559 Ki = 2126 nM T77365 C9AVS8 11952560 Ki = 1656 nM T77365 CD41JX 11952564 Ki = 177 nM T77365 CI6SX1 11952665 Ki = 619 nM T77365 C8OKX0 11952670 Ki = 858 nM T77365 CK3T8W 11953248 Ki = 769 nM T77365 CO29QE 11956192 Ki = 1.6 nM T77365 CM0SL3 11956193 Ki = 2.7 nM T77365 CW8KI0 11956198 Ki = 51 nM T77365 C0KXU5 11977965 Ki > 5000 nM T77365 CXT4S5 11977966 Ki > 5000 nM T77365 CWF2B7 11977967 Ki > 5000 nM T77365 CULI10 11978309 Ki > 5000 nM T77365 C6Z3SF 11978310 Ki > 5000 nM T77365 C1EAC3 11978313 Ki > 5000 nM T77365 CUVN07 11978421 Ki > 5000 nM T77365 C5YU6W 11995348 Ki = 2720 nM T77365 C02DIG 11995349 Ki = 168 nM T77365 CTB21R 11995351 Ki = 2960 nM T77365 C1UGS4 11995353 Ki = 132 nM T77365 CE53IF 11995448 Ki = 1400 nM T77365 C8TD1Y 11995554 Ki = 313 nM T77365 CI1TL9 11995555 Ki = 2260 nM T77365 CUM6T1 11995557 Ki = 681 nM T77365 CF56SH 11995649 Ki > 10000 nM T77365 C8FR7V 11995650 Ki = 7820 nM T77365 C4YPA1 11995651 Ki = 414 nM T77365 CNX94G 12063014 Ki > 10000 nM T77365 CPF9I3 12066874 Ki = 2900 nM T77365 CB7N2Z 12097026 Ki = 1 nM T77365 CWFL86 12267225 Ki = 479 nM T77365 CM04PC 12267228 Ki = 126 nM T77365 CM8B4R 12293993 Ki = 381 nM T77365 C3TJI0 12351799 Ki = 2450 nM T77365 CQ6TX7 12455201 Ki > 10000 nM T77365 CFC36H 12687948 Ki = 52800 nM T77365 C21DPY 12731783 Ki > 5200 nM T77365 CC8Q7D 12766586 Ki = 42300 nM T77365 CTE6H4 13155597 Ki = 460 nM T77365 CWOQ92 13360944 Ki = 42100 nM T77365 CB4M0C 13506474 Ki = 400 nM T77365 C24VJF 13608091 Ki = 145 nM T77365 C97BVY 13830108 Ki = 7 nM T77365 CVS4J0 14426726 Ki = 837 nM T77365 COU82X 14686957 Ki > 10000 nM T77365 CCB92W 14686958 Ki = 5900 nM T77365 CQS35H 14842888 Ki = 519 nM T77365 C76FZJ 14873275 Ki > 10000 nM T77365 CQ7MK8 15388822 Ki = 14700 nM T77365 CSQ0R5 15388827 Ki = 9980 nM T77365 CEN2O9 15388828 Ki = 12200 nM T77365 CPD7A4 15588319 Ki = 7500 nM T77365 C65SCN 15599151 Ki = 2050 nM T77365 C15FWY 15646970 EC50 = 1300 nM T77365 CG0I8D 15667089 Ki = 157 nM T77365 C8OZ5G 15667105 Ki = 980 nM T77365 C4UKS2 15729957 IC50 = 40.74 nM T77365 CE13QR 15729970 Ki = 3.56 nM T77365 CV8DE2 15729973 Ki = 59.1 nM T77365 CFD31U 15729977 Ki = 64.8 nM T77365 C6QT8L 15931307 EC50 = 96200 nM T77365 C5YDU4 15931309 EC50 = 4700 nM T77365 C5BAJ3 15931313 EC50 = 15500 nM T77365 C31TPS 15950360 Ki = 54 nM T77365 C3GP9F 15987727 Ki = 454 nM T77365 C7H5ZS 15987740 Ki = 290 nM T77365 CZUD37 16003546 Ki = 1000 nM T77365 CT9I7F 16036826 Ki = 66 nM T77365 C05KOS 16050635 Ki = 64 nM T77365 CGWF18 16062294 Ki = 40 nM T77365 CI32XZ 16064248 Ki = 4 nM T77365 C6UEW5 16064250 Ki = 259 nM T77365 C6M3VK 16064568 Ki = 76 nM T77365 C04WQF 16064570 Ki = 206 nM T77365 CH72WU 16064711 Ki = 78 nM T77365 C8Z2WO 16070220 Ki = 111 nM T77365 C80TJF 16070335 Ki = 312 nM T77365 CQRU95 16070337 Ki = 312 nM T77365 C8E6CH 16070448 Ki = 312 nM T77365 CWFS63 16071777 Ki = 1.2 nM T77365 C36JRA 16071780 Ki = 879 nM T77365 CX2GC6 16071897 Ki = 1313 nM T77365 C9K2PE 16071901 Ki = 51 nM T77365 CN7F9X 16072019 Ki = 727 nM T77365 CGX62B 16072020 Ki = 55 nM T77365 CL4ON2 16072021 Ki = 44 nM T77365 CU42YH 16072022 Ki = 140 nM T77365 CXS8C0 16072023 Ki = 197 nM T77365 CSO1T2 16072024 Ki = 105 nM T77365 C8W5EP 16087946 Ki > 10000 nM T77365 CA9QY7 16094561 Ki = 6000 nM T77365 C7DV1Q 16094575 Ki = 1800 nM T77365 C1T7DI 16103162 Ki > 5000 nM T77365 C87PRE 16103163 Ki > 5000 nM T77365 C34YIZ 16103164 Ki > 5000 nM T77365 C6U0TL 16103165 Ki = 2100 nM T77365 CT9O5K 16103166 Ki > 5000 nM T77365 CA2W9G 16103167 Ki = 4950 nM T77365 CG74XQ 16103168 Ki = 4100 nM T77365 CL87PX 16103169 Ki = 633 nM T77365 C01PWF 16103170 Ki > 5000 nM T77365 CO3HF4 16103171 Ki > 5000 nM T77365 CIAE42 16103176 Ki = 1550 nM T77365 C0Z4KU 16103177 Ki = 1200 nM T77365 C3Y8IU 16103178 Ki = 1600 nM T77365 CA1EH0 16103179 Ki > 5000 nM T77365 CJ8O9B 16103184 Ki = 3300 nM T77365 CY3R6K 16103185 Ki = 1700 nM T77365 C9F7SM 16103186 Ki = 3800 nM T77365 C7HM0K 16103187 Ki = 3200 nM T77365 CGP93C 16115479 Ki = 3130 nM T77365 CX4O9C 16115613 Ki = 5290 nM T77365 CCZ67Y 16115614 Ki = 18000 nM T77365 C4TDQ5 16115615 Ki = 14700 nM T77365 C4EW6I 16115616 Ki = 18700 nM T77365 C4FI6K 16115617 Ki = 6660 nM T77365 CYKC87 16115749 Ki = 4600 nM T77365 C4A8SU 16115750 Ki = 6290 nM T77365 C8VXL9 16115751 Ki = 12400 nM T77365 CRH54T 16115902 Ki = 12100 nM T77365 C53DBK 16115903 Ki = 16300 nM T77365 CT5UQ7 16115904 Ki = 31700 nM T77365 CRZ0V4 16115905 Ki = 10400 nM T77365 CK87MV 16115906 Ki = 6460 nM T77365 C3G6FA 16115907 Ki = 27100 nM T77365 CC53PW 16116048 Ki = 4210 nM T77365 C0S1VK 16122818 Ki = 5.9 nM T77365 CA49CN 16122819 Ki = 17 nM T77365 COFK82 16128761 Ki = 2.8 nM T77365 C3KXQ7 16202724 Ki = 2570 nM T77365 CFST91 16202843 Ki = 344 nM T77365 C7C3ZJ 16203430 Ki = 2670 nM T77365 CH91QO 16203667 Ki = 277 nM T77365 C4OS0D 16203669 Ki = 250 nM T77365 C0KL4A 16220189 Ki = 341 nM T77365 CZL78O 16344477 Ki > 100000 nM T77365 CZT4J2 16433205 Ki > 100000 nM T77365 CNAX05 16601516 Ki > 100000 nM T77365 C7QI4J 16646020 Ki = 200 nM T77365 C4QU0M 16654984 Ki = 0.4 nM T77365 CFE82W 16656768 Ki > 10000 nM T77365 CO9Q6J 16679348 Ki = 0.9 nM T77365 CH2L3C 16679349 Ki = 0.3 nM T77365 CL8TO3 16679350 Ki = 0.5 nM T77365 C7WF2V 16720104 Ki > 2500 nM T77365 CT7UO9 16720105 Ki > 2500 nM T77365 C9JSW0 16720106 Ki > 2500 nM T77365 C6RT7K 16735280 Ki = 1600 nM T77365 C4VQ5U 16735505 Ki = 4020 nM T77365 C4T9HB 16735540 Ki = 45 nM T77365 CDV52Y 16739249 Ki = 893 nM T77365 CLU01J 16755701 Ki = 11300 nM T77365 C8BL4P 16762757 Ki = 6900 nM T77365 C6PLG1 17035744 Ki = 5.5 nM T77365 CZX1Y3 17035750 Ki = 1.6 nM T77365 C1WAP8 17036152 Ki = 5900 nM T77365 CBR05N 17198004 Ki = 28 nM T77365 C2GR5M 17408222 Ki = 1700 nM T77365 CP0T2V 17427517 Ki = 1000 nM T77365 CWD1N7 17429448 Ki = 300 nM T77365 CTA05E 17487156 Ki = 3400 nM T77365 CUW24Z 17500622 Ki = 2800 nM T77365 C9L0RZ 17517117 Ki = 33000 nM T77365 C1UOA0 17523423 Ki = 6000 nM T77365 CM67RA 17544645 Ki > 100000 nM T77365 COPB05 17562147 Ki > 100000 nM T77365 C0MK3L 17567779 Ki = 13000 nM T77365 C8JYP0 17757368 Ki = 3.1 nM T77365 CXH6D7 17863130 IC50 > 10000 nM T77365 C8BU2E 17863131 IC50 > 10000 nM T77365 CN7D2S 17863136 IC50 > 10000 nM T77365 C41OLX 17863145 IC50 > 650 nM T77365 C72CYF 17863152 IC50 > 10000 nM T77365 CXRL32 17863158 IC50 > 10000 nM T77365 CEM6V1 17863168 IC50 > 10000 nM T77365 C83NVA 17863179 IC50 > 10000 nM T77365 CIJ08G 17863186 IC50 > 10000 nM T77365 CL9AX4 17863209 IC50 > 10000 nM T77365 CELB65 17863210 IC50 > 10000 nM T77365 C6ARU8 17863215 IC50 > 10000 nM T77365 CRH9U4 17863224 IC50 > 10000 nM T77365 COX01L 17863234 IC50 > 10000 nM T77365 CF87SP 18440405 Ki = 27 nM T77365 CX6J0D 18440417 Ki = 14 nM T77365 CRJ31X 18440425 Ki = 150 nM T77365 CKE94U 18440431 Ki = 738 nM T77365 CZO7K8 18440528 Ki = 284 nM T77365 CH29ON 18440555 Ki = 9110 nM T77365 CGT4Q6 18677485 Ki = 14 nM T77365 C1BZ9J 18677506 Ki = 17 nM T77365 CQ6T2X 18677531 Ki = 9 nM T77365 CJ30UR 18677534 Ki = 57 nM T77365 C8M4RO 18677544 Ki = 104 nM T77365 C0VD9T 19574102 Ki = 398.11 nM T77365 CA12QJ 19574107 Ki = 398.11 nM T77365 CBXA48 20592013 Ki = 4590 nM T77365 CZOA41 20605044 Ki = 5.9 nM T77365 CA6K0T 20620151 Ki = 192 nM T77365 C0M7ON 20620157 Ki = 197 nM T77365 CNUH04 20620160 Ki = 23 nM T77365 CPK6Q0 20620161 Ki = 277 nM T77365 CS4GZ0 20759175 Ki = 2420 nM T77365 CBC2U1 20770622 Ki = 1.8 nM T77365 COVH65 20770635 Ki = 1.4 nM T77365 CBJ0O1 20770653 Ki = 1.5 nM T77365 CC2Y8L 20770654 Ki = 2.8 nM T77365 C6U4LK 20770655 Ki = 1.6 nM T77365 C91ICH 20770658 Ki = 5.8 nM T77365 C5KR4S 20847387 Ki > 100000 nM T77365 C1N7ZG 20974732 Ki = 5900 nM T77365 CW50HY 20974734 Ki = 1100 nM T77365 CR2P0O 21054078 Ki > 100000 nM T77365 CM7C5Y 21180383 Ki = 1000 nM T77365 CW53KM 21308711 Ki = 0.03 nM T77365 C6ZWE3 21363898 Ki = 1.5 nM T77365 CFTR39 21363905 Ki = 0.9 nM T77365 CB2V8H 21603068 Ki = 9100 nM T77365 C25WAJ 21874520 Ki = 22 nM T77365 CTK29C 21874538 Ki = 11.9 nM T77365 C96PRF 21874571 Ki = 3.5 nM T77365 C07MZN 21874581 Ki = 5.4 nM T77365 C5QJC8 21874602 Ki = 10.8 nM T77365 CXG16I 21874603 Ki = 2.3 nM T77365 CV2C4F 21874613 Ki = 1.5 nM T77365 CB7S8A 21874626 Ki = 11.1 nM T77365 CKG68C 21874634 Ki = 122 nM T77365 CTX5P2 21874639 Ki = 400 nM T77365 C1CKS9 21874641 Ki = 1.6 nM T77365 CU80AG 21874647 Ki = 2.1 nM T77365 C38CXY 21874661 Ki = 0.7 nM T77365 C4S5PJ 21874662 Ki = 8.6 nM T77365 C14FGO 21874668 Ki = 8.8 nM T77365 C3WLM0 21874675 Ki = 1.1 nM T77365 COLC85 21874676 Ki = 2 nM T77365 C2PZN3 21874681 Ki = 1.6 nM T77365 CP84GK 21874685 Ki = 1.9 nM T77365 CSV0W4 21874686 Ki = 1.5 nM T77365 CW47EF 21874687 Ki = 14.5 nM T77365 C3EK0T 21874692 Ki = 28 nM T77365 C3KH4A 21874697 Ki = 1.9 nM T77365 CDV73C 21874721 Ki = 2.2 nM T77365 C7GWD4 21874722 Ki = 241 nM T77365 C4L8UK 21874755 Ki = 832 nM T77365 CLY0E3 21874756 Ki = 1 nM T77365 CWQ47T 21874764 Ki = 116 nM T77365 C74HIZ 21874771 Ki = 8.5 nM T77365 C7NT1D 21874782 Ki = 2.3 nM T77365 CG9Y7N 21874786 Ki = 3 nM T77365 C7YRN0 21893339 Ki = 572 nM T77365 CK4HL6 21916357 Ki = 3850 nM T77365 CZRX51 21916371 Ki = 633 nM T77365 CS19AF 21916389 Ki = 73 nM T77365 CBY0E6 21916394 Ki = 272 nM T77365 CI1CO9 21916398 Ki = 301 nM T77365 CZ59CO 21916406 Ki = 312 nM T77365 C2XR0J 21916408 Ki = 408 nM T77365 C03FGL 21916419 Ki = 149 nM T77365 CB56UX 21958512 Ki = 217 nM T77365 CBA86P 21958522 Ki > 15000 nM T77365 C4I2HN 21958524 Ki = 2760 nM T77365 CKQ1C3 21958525 Ki > 5000 nM T77365 CBQF27 21958526 Ki = 407 nM T77365 CZ92NC 21958536 Ki = 234 nM T77365 CFX4B6 21958541 Ki = 4910 nM T77365 C2CFG0 21958557 Ki = 125 nM T77365 CZN1L8 21958583 Ki = 139 nM T77365 CW5NK7 21958593 Ki = 1730 nM T77365 C36FJO 21958619 Ki = 234 nM T77365 CJ7IB6 21958676 Ki > 5000 nM T77365 CTSU04 21958681 Ki = 3800 nM T77365 CW5DG9 21958701 Ki = 1500 nM T77365 C7RE2I 21958724 Ki = 247 nM T77365 CJO62E 21958725 Ki = 3400 nM T77365 C6F8TR 21958745 Ki > 5000 nM T77365 CMF03Z 21958758 Ki = 3000 nM T77365 C58MPT 21958761 Ki > 5000 nM T77365 C5L8YT 21958762 Ki = 496 nM T77365 C4K7OP 21958764 Ki = 261 nM T77365 CCTJ56 21958775 Ki = 100 nM T77365 CU7EZ3 21958783 Ki > 5000 nM T77365 CUNF42 21958814 Ki = 3400 nM T77365 C5HFL6 22002319 Ki = 25.8 nM T77365 CFH75K 22002352 Ki = 5320 nM T77365 C02SLQ 22002364 Ki = 116 nM T77365 CPS61Y 22002375 Ki = 15 nM T77365 C3CV9X 22002449 Ki = 3.32 nM T77365 CW24GQ 22015484 Ki = 16 nM T77365 CEWY38 22015485 Ki = 6 nM T77365 CNJ90S 22015489 Ki = 4 nM T77365 CDUS06 22015491 Ki = 1322 nM T77365 C8M3PX 22015492 Ki = 2086 nM T77365 CDN7B6 22015493 Ki = 9 nM T77365 C6P2DA 22015494 Ki = 110 nM T77365 CD0KT8 22015499 Ki = 4 nM T77365 CJ0Z6F 22015500 Ki = 48 nM T77365 CN7O2U 22015504 Ki = 1 nM T77365 C05CGK 22015508 Ki = 8 nM T77365 CQ07MJ 22015509 Ki = 17 nM T77365 CG8Z5Y 22015516 Ki = 9 nM T77365 CV6F4T 22015525 Ki = 135 nM T77365 C48YPI 22015526 Ki = 119 nM T77365 CQL6X2 22015529 Ki = 1891 nM T77365 CS8IX9 22015530 Ki = 4 nM T77365 C7RV4D 22015532 Ki = 1 nM T77365 CVH03D 22015533 Ki = 36 nM T77365 CYN5L0 22015535 Ki = 26 nM T77365 CU41EO 22015539 Ki = 1616 nM T77365 CAU0Z3 22015549 Ki = 45 nM T77365 CPK81R 22015550 Ki = 3 nM T77365 CKME84 22055296 Ki = 16 nM T77365 C43TSO 22055299 Ki = 10 nM T77365 CE6U0L 22220610 Ki = 44.3 nM T77365 C67RYE 22252243 Ki = 25 nM T77365 C7CW3I 22266730 Ki > 5000 nM T77365 CZF4S2 22266732 Ki > 5000 nM T77365 CTO91Z 22266738 Ki = 1200 nM T77365 C75PVI 22266740 Ki > 5000 nM T77365 CC2N6M 22266741 Ki > 5000 nM T77365 CZL43T 22266742 Ki > 5000 nM T77365 C0XT6H 22266744 Ki = 1220 nM T77365 CV6E4A 22266746 Ki = 73 nM T77365 CU16OK 22266751 Ki > 5000 nM T77365 C2QUH0 22266756 Ki > 5000 nM T77365 CLF81K 22266759 Ki > 5000 nM T77365 CIOB39 22266761 Ki > 5000 nM T77365 CC12SJ 22266763 Ki = 2700 nM T77365 C4ZJ1F 22266765 Ki = 1800 nM T77365 C3WK8Z 22266766 Ki > 5000 nM T77365 CAGC71 22266769 Ki = 2370 nM T77365 CV53YM 22266771 Ki > 5000 nM T77365 CSC37U 22266775 Ki = 420 nM T77365 CCQ0I1 22266776 Ki > 5000 nM T77365 CDWI49 22266778 Ki = 481 nM T77365 CC94DE 22266784 Ki > 5000 nM T77365 C7G0LF 22282339 Ki > 826 nM T77365 CPDA63 22283414 Ki = 250 nM T77365 CW8B7M 22422193 Ki = 1584.89 nM T77365 CA6M3I 22517807 Ki = 5100 nM T77365 CYP2Z4 22674365 Ki = 16 nM T77365 CL95BF 22674372 Ki = 29 nM T77365 CIHV23 22674379 Ki = 92 nM T77365 CIK25F 22674386 Ki = 80 nM T77365 CJVG74 22674390 Ki = 4.3 nM T77365 CJ1H3A 22674393 Ki = 56 nM T77365 CXV1G4 22674398 Ki = 22 nM T77365 CV3IJ9 22674410 Ki = 25 nM T77365 C0ITC9 22674411 Ki = 8.1 nM T77365 CQ16FW 22674422 Ki = 3055 nM T77365 C54ZKH 22674428 Ki = 60 nM T77365 CZS72H 22674456 Ki = 49 nM T77365 C4PK7T 22674477 Ki = 25 nM T77365 CE7FI3 22674484 Ki = 335 nM T77365 C1T3OA 22674492 Ki = 118 nM T77365 CJ52EV 23371936 Ki > 100000 nM T77365 CFT0A1 23371944 Ki > 100000 nM T77365 CIV69F 23438858 Ki = 190 nM T77365 C8XRA5 23540117 Ki = 0.7 nM T77365 C3Y7PK 23540125 Ki = 2.5 nM T77365 CODM62 23540126 Ki = 40 nM T77365 CEW7T3 23540131 Ki = 25 nM T77365 C6OCL1 23546899 Ki = 28 nM T77365 CPC5N2 23552495 Ki = 5 nM T77365 CP10SH 23570387 Ki = 0.5 nM T77365 C65SJK 23656931 Ki = 20.1 nM T77365 CGRT64 23656932 Ki = 50.6 nM T77365 C8N0LF 23656933 Ki = 67.5 nM T77365 CYU94Z 23656934 Ki = 1030 nM T77365 C8SC3A 23656935 Ki > 10000 nM T77365 CO98NZ 23656936 Ki > 10000 nM T77365 CV28WL 23656937 Ki > 10000 nM T77365 CAG3Y8 23657103 Ki = 4800 nM T77365 CKRG98 23657104 Ki = 262.1 nM T77365 C6YS2Z 23657105 Ki = 134 nM T77365 CZ6H4G 23657106 Ki = 493.3 nM T77365 C6F4UV 23657107 Ki = 9 nM T77365 C26AWG 23657108 Ki = 4.7 nM T77365 C0R9DW 23657109 Ki = 2.3 nM T77365 COD51S 23657262 Ki > 10000 nM T77365 CSZB58 23657263 Ki > 10000 nM T77365 C68QBD 23657264 Ki > 10000 nM T77365 C1SWM6 23657265 Ki > 10000 nM T77365 CG4I1H 23657266 Ki > 10000 nM T77365 CMSG38 23657267 Ki = 460.2 nM T77365 C6GDP9 23657408 Ki = 625 nM T77365 CVBI12 23657409 Ki = 120.1 nM T77365 CFE2N1 23757284 Ki = 2 nM T77365 CVO53U 23900137 Ki = 39 nM T77365 C1M0YR 24699001 Ki = 10000 nM T77365 CG8BZ4 24739307 Ki = 0.3 nM T77365 C1SGW5 24739308 Ki = 1 nM T77365 CFVO28 24739309 Ki = 0.3 nM T77365 CU12PX 24739310 Ki = 0.2 nM T77365 CK96FD 24739478 Ki = 0.3 nM T77365 CJ23NC 24739479 Ki = 5.7 nM T77365 CUW7F4 24739481 Ki = 0.9 nM T77365 CG95TO 24739646 Ki = 0.3 nM T77365 C5JK9I 24739647 Ki = 1.2 nM T77365 CO46JZ 24739648 Ki = 0.5 nM T77365 CQ5H6Y 24739649 Ki = 2.3 nM T77365 COB5Q7 24739812 Ki = 0.5 nM T77365 C1Y7AV 24739813 Ki = 1.4 nM T77365 CRN05P 24739814 Ki = 0.5 nM T77365 CRT41U 24768400 Ki = 0.9 nM T77365 C3EVZ7 24768401 Ki = 2 nM T77365 CIU04J 24768402 Ki = 135 nM T77365 C8I3OV 24768403 Ki = 14 nM T77365 C7RGV4 24768404 Ki = 12 nM T77365 C2PRD9 24768405 Ki = 24 nM T77365 CS7M9E 24768406 Ki = 131 nM T77365 C3NO0Z 24768407 Ki = 27 nM T77365 CJD61X 24768408 Ki = 1000 nM T77365 C5X9OD 24768409 Ki = 190 nM T77365 CF6BC7 24768410 Ki = 17 nM T77365 CAG7S1 24768411 Ki = 53.4 nM T77365 CAG8R2 24768412 Ki = 25.5 nM T77365 CSL71N 24768413 Ki = 9 nM T77365 CJ2V9Z 24768414 Ki = 11 nM T77365 CZ4J5K 24768415 Ki = 10 nM T77365 CQ63KX 24768416 Ki = 10 nM T77365 C8OGP3 24768417 Ki = 1.5 nM T77365 C4ZRC9 24768418 Ki = 2.9 nM T77365 C1A0NS 24768419 Ki = 3.6 nM T77365 C35QUL 24768420 Ki = 5.7 nM T77365 C6XR5O 24768421 Ki = 6 nM T77365 CAG3S6 24768422 Ki = 15 nM T77365 CI6B4H 24768423 Ki = 5.4 nM T77365 CXEC07 24768424 Ki = 8.6 nM T77365 CS0C6Q 24768425 Ki = 3.7 nM T77365 C3E6MK 24768426 Ki = 4 nM T77365 C46NSY 24768427 Ki = 86 nM T77365 CF8C0L 24768428 Ki = 3.8 nM T77365 CBMC42 24768429 Ki = 2.5 nM T77365 CR5H8A 24768430 Ki = 4.4 nM T77365 CA3UK5 24768431 Ki = 11 nM T77365 CG8QK3 24768432 Ki = 2.1 nM T77365 CMT5N1 24768433 Ki = 2.1 nM T77365 C6HW8J 24768434 Ki = 2.4 nM T77365 CEA0J5 24768437 Ki = 1121 nM T77365 C8NKT5 24768438 Ki = 398 nM T77365 CGVO15 24768442 Ki = 71 nM T77365 C53BPO 24768445 Ki = 4149 nM T77365 C6ZDA2 24778159 Ki = 5.2 nM T77365 C9OY1E 24779894 Ki = 439 nM T77365 C53LCQ 24779896 Ki = 2380 nM T77365 C40ZDL 24779898 Ki = 4710 nM T77365 C5B0ZH 24781767 Ki = 17 nM T77365 CP0JB3 24781768 Ki = 46 nM T77365 CXU4L5 24781917 Ki = 48 nM T77365 CCT1V7 24781918 Ki = 48 nM T77365 C7KS3N 24782079 Ki = 210 nM T77365 C2BV7I 24803315 Ki = 382 nM T77365 C6S1HG 24810000 Ki = 1.8 nM T77365 CK02ZF 24812771 Ki = 4.7 nM T77365 C5UO3Z 24827415 Ki = 2050 nM T77365 C32BCU 24827417 Ki = 1150 nM T77365 CKC0W3 24827442 Ki = 1090 nM T77365 C0WA2D 24827443 Ki = 411 nM T77365 CQW7H1 24827444 Ki = 312 nM T77365 CIR6E9 24827552 Ki = 670 nM T77365 C15VIG 24827553 Ki = 2250 nM T77365 C06PBV 24827554 Ki = 5410 nM T77365 C34RNS 24827555 Ki = 2280 nM T77365 CGUY42 24827556 Ki = 1950 nM T77365 C2W7YS 24828056 Ki = 1390 nM T77365 CWPS95 24828457 Ki = 2500 nM T77365 CU0Q2I 24878975 Ki > 10000 nM T77365 C05BYL 24882472 Ki = 8760 nM T77365 C8DTC3 24894065 Ki = 2.4 nM T77365 C0PHN9 24939231 Ki = 159 nM T77365 C0WF2D 24950372 Ki = 140 nM T77365 C47TZM 24950529 Ki = 190 nM T77365 CY5W4G 24950531 Ki = 41 nM T77365 C31DGI 24950532 Ki = 92 nM T77365 CU24RD 24950533 Ki = 26 nM T77365 C45DXE 24950690 Ki = 140 nM T77365 C6PT5O 24950691 Ki = 58 nM T77365 CL6T3O 24950845 Ki = 640 nM T77365 CS1ZM6 24950846 Ki = 15 nM T77365 CZK1X7 24989636 Ki = 12 nM T77365 CWPX23 24989637 Ki = 110 nM T77365 C03WIO 24989638 Ki = 261 nM T77365 CPD0U1 24989640 Ki = 69 nM T77365 C0YGQ2 24998410 Ki = 10100 nM T77365 C2EK5G 25002987 Ki = 1260 nM T77365 COSA97 25003338 Ki = 440 nM T77365 C7DF0O 25003339 Ki = 420 nM T77365 C1ZXW0 25003340 Ki = 230 nM T77365 CL5NI4 25008276 IC50 >= 10000 nM T77365 CW5YA6 25066016 Ki = 3.3 nM T77365 CX43GT 25069599 Ki = 87 nM T77365 CP3Y5K 25069603 Ki = 7.9 nM T77365 CM1WB9 25069914 Ki = 0.83 nM T77365 CK92QL 25070230 Ki = 316.23 nM T77365 C04QRE 25074004 Ki = 0.72 nM T77365 C07GFA 25074313 Ki = 3 nM T77365 CLWN54 25074316 Ki = 0.4 nM T77365 CWFC39 25104832 Ki = 280 nM T77365 CAX68Y 25104834 Ki = 167 nM T77365 CMX24U 25110630 Ki = 1 nM T77365 C7I9MV 25110821 Ki = 1 nM T77365 C3YH5W 25138072 Ki = 87 nM T77365 CMP7V1 25138073 Ki = 120 nM T77365 CLW7O5 25138074 Ki = 40 nM T77365 C7L6SP 25138075 Ki = 0.92 nM T77365 C1PF5O 25138076 Ki = 0.6 nM T77365 CC4HW2 25138077 Ki = 0.19 nM T77365 C9J1MQ 25138078 Ki = 2.3 nM T77365 C9LMW0 25138079 Ki = 2.9 nM T77365 C2QLK4 25138080 Ki = 3.1 nM T77365 CS89DE 25138081 Ki = 4 nM T77365 C5AJ0V 25138082 Ki = 1.8 nM T77365 CAL52B 25138083 Ki = 7.4 nM T77365 CZ41XS 25138084 Ki = 7.8 nM T77365 CA7JE4 25138085 Ki = 12 nM T77365 C9GZ6D 25138086 Ki = 0.61 nM T77365 C5A1FW 25138087 Ki = 0.26 nM T77365 CZ49VH 25138088 Ki = 0.56 nM T77365 CA01RE 25138089 Ki = 2.3 nM T77365 CC5O4P 25138090 Ki = 0.71 nM T77365 CQ30KW 25138091 Ki = 0.47 nM T77365 CCM9X1 25138092 Ki = 1.9 nM T77365 C7JE1V 25147618 Ki > 1000 nM T77365 C5FHU3 25147619 Ki > 1000 nM T77365 CN2FL7 25188209 Ki = 41 nM T77365 CB6QZ9 25207803 IC50 = 965 nM T77365 C1O2VJ 25207955 Ki = 4.2 nM T77365 CD2BJ5 25207956 Ki = 28 nM T77365 C5J0UG 25207957 Ki = 205 nM T77365 CIVO18 25207958 Ki > 10000 nM T77365 C5ZHT9 25207959 Ki = 9 nM T77365 C1YWI8 25207960 Ki = 324 nM T77365 CJ8LD2 25207961 Ki = 455 nM T77365 CHT85D 25208107 Ki = 40 nM T77365 CL7UJ3 25208108 Ki = 439 nM T77365 CL5JR6 25208109 Ki = 7.5 nM T77365 C8RW4K 25208254 Ki = 23 nM T77365 CXK1G5 25208255 Ki = 119 nM T77365 CR6O3B 25208256 Ki = 27 nM T77365 CA3LY1 25208257 Ki = 20 nM T77365 C6TI7Y 25208258 Ki = 46 nM T77365 C2WT8G 25208259 Ki = 5.9 nM T77365 CN9XE6 25208260 Ki = 19 nM T77365 CHG1N9 25209990 Ki = 50 nM T77365 C0IBC5 25209991 Ki = 2.7 nM T77365 CFT98K 25210116 Ki = 47 nM T77365 CYK7O5 25210117 Ki = 15 nM T77365 CEYP97 25210118 Ki = 50 nM T77365 CZ3E6O 25210119 Ki = 43 nM T77365 C7MI5W 25210254 Ki = 92 nM T77365 C74JQH 25210255 Ki = 78 nM T77365 COF2H0 25210256 Ki = 313 nM T77365 C7T6PR 25210257 Ki = 1867 nM T77365 CI01GB 25211166 Ki = 88 nM T77365 CU6OR2 25211167 Ki = 43 nM T77365 CJ0S1U 25230098 IC50 = 7107 nM T77365 CN3QA7 25230100 IC50 = 3093 nM T77365 CJO09C 25230180 IC50 = 6760 nM T77365 C5PT8L 25230181 IC50 = 468 nM T77365 CH61DM 25230881 IC50 = 1417 nM T77365 CE4GZ7 25230948 IC50 = 2485 nM T77365 C8W0PI 25230949 IC50 > 10000 nM T77365 CCJ16P 25231166 IC50 = 2347 nM T77365 C6C5EJ 25231167 IC50 = 2516 nM T77365 C3N2CW 25231168 IC50 = 6136 nM T77365 CV4CT2 25231169 IC50 = 710 nM T77365 CUI20F 25231170 IC50 = 2610 nM T77365 C6S0OK 25242240 Ki = 0.3 nM T77365 CJ4K1Z 25242440 Ki = 8.2 nM T77365 CI1GW6 25268841 Ki = 6.5 nM T77365 C0Z5KG 25392045 Ki > 100000 nM T77365 CY18BR 25573285 Ki = 200 nM T77365 CS0V9B 32178888 Ki = 1000 nM T77365 C8DT0B 32459044 Ki = 1400 nM T77365 CJ95TD 32459103 Ki = 3900 nM T77365 CFW2X3 32459568 Ki = 6400 nM T77365 CSE07H 32459683 Ki = 1700 nM T77365 C4MB8S 32460014 Ki = 2200 nM T77365 C3FH2I 32460336 Ki = 1000 nM T77365 C6LI7R 32460717 Ki = 200 nM T77365 C7Z2BV 32460731 Ki = 2500 nM T77365 C01BKR 32460889 Ki = 1800 nM T77365 C6VG3H 32461058 Ki = 8800 nM T77365 CU51PG 32461094 Ki = 2000 nM T77365 C4OUE0 32461100 Ki = 3200 nM T77365 C8TE4D 32461405 Ki = 1000 nM T77365 CKS89N 32461556 Ki = 4000 nM T77365 C40SYI 32866639 Ki = 2900 nM T77365 CZF25S 40041829 Ki = 1200 nM T77365 CXK0H7 41316339 Ki > 100000 nM T77365 CWUA82 42625614 Ki > 100000 nM T77365 C6W4XM 42625615 Ki = 16200 nM T77365 CX8DV9 42625691 Ki > 100000 nM T77365 C5I8NE 42625766 Ki = 2190 nM T77365 CIG29P 42625767 Ki > 100000 nM T77365 CETQ95 42626002 Ki = 211 nM T77365 CBW7G5 42626003 Ki = 208 nM T77365 C6RIC7 42626004 Ki = 2240 nM T77365 C8RDW2 42626220 Ki = 208 nM T77365 C4RHY0 42630191 IC50 = 5050 nM T77365 CDSI21 42631399 Ki = 1100 nM T77365 C5YV2R 42631400 Ki = 1000 nM T77365 CP31OD 42631506 Ki = 600 nM T77365 CKEC01 42631507 Ki = 100 nM T77365 CBJ07K 42631609 Ki = 400 nM T77365 C1QS2X 42631610 Ki = 1400 nM T77365 CVX80U 42631613 Ki = 600 nM T77365 C6SVP2 42631614 Ki = 700 nM T77365 C0O1HM 42631715 Ki = 100000 nM T77365 C3M5GK 42631719 Ki = 400 nM T77365 C0EYB8 42631813 Ki = 2700 nM T77365 C0UH7I 42631818 Ki = 100 nM T77365 CT57MJ 42631819 Ki = 800 nM T77365 CS0O4J 42631924 Ki = 400 nM T77365 CTBW80 42636897 Ki = 1340 nM T77365 CK43JX 44157013 Ki = 9 nM T77365 C1J6SG 44185870 Ki = 48.4 nM T77365 CX24EI 44185874 Ki = 3720 nM T77365 CWX1B7 44185933 Ki = 271 nM T77365 C8I9LD 44185936 Ki = 94.5 nM T77365 CQRH91 44186579 Ki = 152 nM T77365 C9RG0P 44186580 Ki = 6.49 nM T77365 CCNH98 44186622 Ki = 161 nM T77365 CY2D4F 44186623 Ki = 92 nM T77365 CAY95F 44186625 Ki = 144 nM T77365 C42DUI 44186626 Ki = 278 nM T77365 CYE0X8 44186667 Ki = 145 nM T77365 CM7B3X 44186668 Ki = 69.4 nM T77365 C69VCO 44186669 Ki = 306 nM T77365 C5X9NC 44186716 Ki = 236 nM T77365 C6JG3Q 44186717 Ki = 328 nM T77365 CE21OP 44186718 Ki = 102 nM T77365 C9W0OQ 44186719 Ki = 112 nM T77365 CE2IV7 44199445 Ki = 0.5 nM T77365 CE6C9F 44203644 Ki = 4568 nM T77365 CFR8Z7 44216394 Ki = 0.8 nM T77365 CZL80X 44216395 Ki = 0.7 nM T77365 C3DW4Q 44217535 Ki = 636 nM T77365 C6I4TU 44217536 Ki = 14.2 nM T77365 C4N2ZM 44217687 Ki = 10.5 nM T77365 C5SK0H 44217688 Ki = 11 nM T77365 C3AE2U 44217689 Ki = 12.7 nM T77365 CH2J3B 44217690 Ki = 12.9 nM T77365 C4KT5J 44217845 Ki = 791 nM T77365 C3CBK6 44217846 Ki = 0.3 nM T77365 CXZI71 44217847 Ki = 0.4 nM T77365 CLG0R9 44218006 Ki = 6.7 nM T77365 CQ90HW 44218008 Ki = 8.9 nM T77365 CW4H8L 44218164 Ki = 9 nM T77365 C8CV9A 44218166 Ki = 23.4 nM T77365 CKZU79 44218167 Ki = 27.4 nM T77365 C47CIO 44218168 Ki = 28.4 nM T77365 CG5BH8 44218327 Ki = 5.2 nM T77365 C3DOH6 44218330 Ki = 381 nM T77365 CC35JG 44219683 Ki = 97.72 nM T77365 CXIT13 44219684 Ki = 112.2 nM T77365 CK1H5B 44241696 Ki = 164 nM T77365 C7T0ZY 44281663 Ki > 1000 nM T77365 CX3YV9 44281684 Ki > 1000 nM T77365 CJ3QM8 44281700 Ki > 1000 nM T77365 CN72HK 44281738 Ki > 1000 nM T77365 C7HV4D 44284007 Ki = 10800 nM T77365 CL8XS1 44284052 Ki = 1940 nM T77365 C28QCM 44284065 Ki = 1780 nM T77365 C8YHM6 44284095 Ki = 4570 nM T77365 CUR2Q6 44284189 Ki = 2410 nM T77365 CE5V1M 44284209 Ki = 2180 nM T77365 CBQ90F 44284222 Ki = 2000 nM T77365 C34FVI 44284223 Ki = 7750 nM T77365 CT0EV8 44284345 Ki = 4100 nM T77365 CCQ4Y0 44317558 Ki = 1136 nM T77365 CW93LX 44317576 Ki = 811 nM T77365 CW1G8S 44317578 Ki = 215 nM T77365 C1RFW2 44317916 Ki = 962 nM T77365 CJS3C0 44317969 IC50 = 3218 nM T77365 C8T0GE 44327984 Ki = 1800 nM T77365 CGF8E6 44330651 Ki > 100000 nM T77365 C4D3VP 44330661 Ki > 100000 nM T77365 CQM47G 44330671 Ki > 100000 nM T77365 C9HCX7 44330672 Ki > 100000 nM T77365 CD1X0S 44330675 Ki > 100000 nM T77365 C2ZM8Y 44330685 Ki > 100000 nM T77365 CEM2V6 44330697 Ki = 6680 nM T77365 C47YKV 44330734 Ki = 880 nM T77365 CB81AF 44330735 Ki > 100000 nM T77365 CNE3L7 44330736 Ki > 100000 nM T77365 C74RDN 44330758 Ki = 1660 nM T77365 C2YS4M 44330775 Ki = 3430 nM T77365 CX50ZN 44330776 Ki > 100000 nM T77365 CA8G4N 44330792 Ki = 5900 nM T77365 C0C4ZU 44330810 Ki > 100000 nM T77365 CZ1E4Q 44330818 Ki = 10000 nM T77365 C4W8MJ 44330819 Ki > 100000 nM T77365 CU6IF4 44330820 Ki = 1710 nM T77365 CR56XK 44330838 Ki > 100000 nM T77365 CSUD59 44330852 Ki = 380 nM T77365 C8J6CZ 44330870 Ki = 120 nM T77365 CX6A2R 44331905 Ki = 4500 nM T77365 CN4PJ9 44331907 Ki = 49000 nM T77365 C2L0JD 44331997 Ki = 13500 nM T77365 C2WU1X 44333135 Ki > 10000 nM T77365 C6ALX7 44333187 Ki > 10000 nM T77365 CVGR26 44333267 Ki > 10000 nM T77365 C1SVU5 44333456 Ki > 10000 nM T77365 CGTS60 44333467 Ki > 10000 nM T77365 CZVN76 44340390 Ki = 61 nM T77365 CN4U6M 44352986 Ki = 0.16 nM T77365 CY2ED1 44352987 Ki = 6.2 nM T77365 CFO54N 44352988 Ki = 36 nM T77365 CM0T9J 44353004 Ki = 2.2 nM T77365 C21TGS 44353021 Ki = 85 nM T77365 CNZ28O 44353022 Ki = 1.8 nM T77365 CZIS51 44353044 Ki = 39 nM T77365 CNE2K6 44353045 Ki = 0.1 nM T77365 CHS5M2 44353053 Ki = 25 nM T77365 CG3PQ9 44353177 Ki = 171 nM T77365 CA1HT6 44353188 Ki = 0.08 nM T77365 COTG37 44353321 Ki = 0.8 nM T77365 CE0GW9 44379809 Ki = 40 nM T77365 CAR18K 44379832 Ki = 100 nM T77365 CLU60V 44379847 Ki = 10 nM T77365 C80YID 44379848 Ki = 1000 nM T77365 CF5DW6 44379908 Ki = 80 nM T77365 CB37DU 44379941 Ki = 5 nM T77365 CJ6ZS4 44379943 Ki > 5200 nM T77365 CE0ZW7 44379970 Ki > 5200 nM T77365 C9BV7F 44379976 Ki = 700 nM T77365 CEQ85H 44379977 Ki = 100 nM T77365 CX37RK 44380025 Ki = 400 nM T77365 CODH02 44380101 Ki = 70 nM T77365 CP9R3J 44380104 Ki = 20 nM T77365 C4I3HP 44380110 Ki = 20 nM T77365 C53IPV 44380120 Ki = 700 nM T77365 CT58NY 44380141 Ki = 2000 nM T77365 C7CJ3S 44380142 Ki = 1200 nM T77365 CHA69W 44380242 Ki = 100 nM T77365 CSRH15 44380243 Ki = 90 nM T77365 CW3E2X 44380262 Ki = 60 nM T77365 C0AIN9 44387759 Ki = 4.3 nM T77365 CC02XN 44388218 Ki = 288 nM T77365 C1T2FP 44388225 Ki = 297 nM T77365 CY4DQ7 44390444 Ki > 5000 nM T77365 C3D6LX 44390522 Ki > 5000 nM T77365 CF6WX2 44390523 Ki = 1010 nM T77365 C25RFG 44390527 Ki > 5000 nM T77365 CWR5M2 44390528 Ki > 5000 nM T77365 CBZ2P1 44390545 Ki > 23 nM T77365 CEB5I3 44390547 Ki > 5000 nM T77365 CE53OI 44390549 Ki > 5000 nM T77365 CG4KO6 44390551 Ki > 5000 nM T77365 CHZ5D1 44390559 Ki = 3140 nM T77365 C6HBX7 44390571 Ki > 5000 nM T77365 C6XV9J 44390583 Ki > 5000 nM T77365 CLQ41H 44390587 Ki > 5000 nM T77365 CA4KL8 44390599 Ki > 5000 nM T77365 C0XIJ4 44390615 Ki > 5000 nM T77365 CD2F9O 44390651 Ki > 5000 nM T77365 C8Q9XH 44390669 Ki > 5000 nM T77365 C4PZC8 44394688 Ki = 1.3 nM T77365 CH5O6U 44394716 Ki = 0.33 nM T77365 C83KXG 44396444 Ki > 5000 nM T77365 C7K1ST 44396450 Ki > 5000 nM T77365 C4AOY9 44396470 Ki > 3900 nM T77365 C32JTS 44396478 Ki = 4100 nM T77365 CHY08U 44396487 Ki = 4000 nM T77365 CS0D8B 44396500 Ki = 4000 nM T77365 C8B1XJ 44396515 Ki > 5000 nM T77365 CXZ7Q4 44396516 Ki = 52 nM T77365 CY7B3D 44396545 Ki > 4000 nM T77365 C7ERK1 44396546 Ki = 3300 nM T77365 C0N1FZ 44396599 Ki > 5000 nM T77365 C4TU8O 44397776 Ki = 39000 nM T77365 C4QNR0 44401051 Ki = 2300 nM T77365 CXCE96 44401487 Ki = 2500 nM T77365 C5U2YX 44401545 Ki = 2300 nM T77365 C8HO4J 44401558 Ki = 3.1 nM T77365 C63DYM 44401720 Ki = 381 nM T77365 CYI29X 44401735 Ki = 22 nM T77365 CM31GR 44401764 Ki = 26 nM T77365 CA10TM 44401805 Ki = 21.5 nM T77365 CC8J5F 44401808 Ki = 7.1 nM T77365 C48JOM 44401809 Ki = 5.6 nM T77365 C9NS2O 44401884 Ki = 7.7 nM T77365 CB6TF9 44401899 Ki = 6.3 nM T77365 CQB9N1 44401992 Ki = 8.7 nM T77365 CXHS76 44402758 Ki = 5610 nM T77365 CV8BG5 44402784 Ki = 175 nM T77365 CFR09M 44403549 Ki = 7140 nM T77365 CDX4H0 44403550 Ki = 870 nM T77365 C14IUF 44403555 Ki = 500 nM T77365 CK2NB5 44403556 Ki = 160 nM T77365 C7WY6E 44403562 Ki = 6780 nM T77365 CQ02SL 44403563 Ki > 10000 nM T77365 C0EYI9 44403568 Ki = 67 nM T77365 C9XJQ4 44403569 Ki = 3543 nM T77365 C0GYJ4 44403586 Ki > 10000 nM T77365 CWQ41V 44403587 Ki > 10000 nM T77365 C3QA1H 44403590 Ki > 10000 nM T77365 C7MA2P 44403595 Ki = 57 nM T77365 CGYE73 44403596 Ki > 10000 nM T77365 C8QT7Y 44403599 Ki > 10000 nM T77365 CB89RY 44403600 Ki = 720 nM T77365 C6MWR3 44403601 Ki = 980 nM T77365 C1Z9AL 44403602 Ki = 1169 nM T77365 CE25OU 44403603 Ki > 10000 nM T77365 CZW73B 44403608 Ki > 10000 nM T77365 CR06AD 44403609 Ki = 30 nM T77365 COKU07 44403611 Ki = 8660 nM T77365 C5CZ7U 44403618 Ki = 1750 nM T77365 C5WED3 44403621 Ki = 830 nM T77365 C4C1WB 44403622 Ki = 360 nM T77365 CMYR63 44403623 Ki = 640 nM T77365 CU1BD7 44403629 Ki = 115 nM T77365 C3EF0B 44403630 Ki = 740 nM T77365 CV16HJ 44403635 Ki = 159 nM T77365 CK73CA 44403636 Ki = 140 nM T77365 CG5HM3 44403643 Ki = 35 nM T77365 CA54QX 44403644 Ki = 115 nM T77365 CP1LQ8 44403649 Ki = 99 nM T77365 CG4UW8 44403654 Ki = 146 nM T77365 C96LYT 44403660 Ki = 1644 nM T77365 CI72ZU 44403661 Ki = 588 nM T77365 CS41TF 44405057 Ki = 4900 nM T77365 CTE46U 44405094 Ki > 10000 nM T77365 CB3X0L 44405124 Ki = 720 nM T77365 CN94AX 44406328 Ki > 5000 nM T77365 C3JPG9 44406334 Ki > 5000 nM T77365 C3S9CP 44406397 Ki > 5000 nM T77365 CAF1Y3 44406398 Ki > 5000 nM T77365 CT21RA 44406403 Ki > 5000 nM T77365 CA8FV4 44406545 Ki = 2500 nM T77365 CG8MQ9 44406555 Ki = 1600 nM T77365 CUPC05 44406556 Ki > 5000 nM T77365 C5ZW8S 44406562 Ki > 5000 nM T77365 CQ98MC 44406567 Ki > 5000 nM T77365 CN7V0Y 44406570 Ki > 5000 nM T77365 CI19OT 44406582 Ki > 5000 nM T77365 CZPM65 44406588 Ki > 5000 nM T77365 C6O9TH 44406592 Ki > 5000 nM T77365 CJA23V 44406607 Ki = 2500 nM T77365 CV5AO7 44406611 Ki > 5000 nM T77365 CE3CP9 44406617 Ki > 5000 nM T77365 CVQ2B8 44406625 Ki > 5000 nM T77365 CD9E7F 44406639 Ki > 5000 nM T77365 CK7GF1 44406642 Ki > 5000 nM T77365 CPEV01 44406643 Ki > 5000 nM T77365 C9ZY1L 44406891 Ki = 79.43 nM T77365 CXL90H 44406904 Ki > 1000 nM T77365 CR8AU6 44406906 Ki = 165.96 nM T77365 CTHP76 44406920 Ki = 10.96 nM T77365 C9XF6Y 44406930 Ki = 2.138 nM T77365 CK9ZB7 44407518 Ki > 10000 nM T77365 CES29R 44408316 Ki = 110 nM T77365 C0EB9D 44410399 Ki = 6707 nM T77365 C6E4RA 44410402 Ki = 935 nM T77365 C5IVA3 44410403 Ki = 344 nM T77365 CI7W8R 44410406 Ki = 59.3 nM T77365 CWQX21 44410409 Ki = 497 nM T77365 CJ26LR 44410410 Ki = 7350 nM T77365 CG30RK 44410412 Ki = 571 nM T77365 CK8I1V 44410544 Ki = 1107 nM T77365 CO2LJ0 44410545 Ki = 642 nM T77365 CX9OZ0 44410549 Ki = 2433 nM T77365 C7DER1 44410550 Ki = 371 nM T77365 C6E8OT 44410551 Ki = 2130 nM T77365 CZ94PN 44410554 Ki = 401 nM T77365 COWL13 44410555 Ki = 645 nM T77365 CHU6Q0 44410556 Ki = 785 nM T77365 CVYF89 44410559 Ki = 3783 nM T77365 C2YF8L 44410561 Ki = 143 nM T77365 CXD2R9 44410566 Ki = 207 nM T77365 C20FJQ 44410585 Ki = 321 nM T77365 CQ8E2B 44410597 Ki = 711 nM T77365 CYG5K3 44410655 Ki = 543 nM T77365 C8DE9A 44410690 Ki = 680 nM T77365 CSTP07 44410691 Ki = 467 nM T77365 CV37TH 44410697 Ki = 152 nM T77365 COD4F9 44417680 Ki = 1660 nM T77365 CM10LW 44420100 Ki = 23 nM T77365 CND70C 44420101 Ki = 31 nM T77365 CSR4Q2 44420921 Ki = 10.9 nM T77365 CWJ19B 44420922 Ki = 13.3 nM T77365 CO68UH 44420926 Ki = 628 nM T77365 CUE35G 44420928 Ki = 413 nM T77365 C1V0HC 44420930 Ki = 58.1 nM T77365 C01VYU 44420931 Ki = 69.3 nM T77365 C3C8LS 44423811 Ki > 1000 nM T77365 CWCH32 44423812 Ki > 1000 nM T77365 CDY6P7 44423813 Ki > 1000 nM T77365 CYR14N 44423814 Ki > 1000 nM T77365 C2F3DE 44423815 Ki > 1000 nM T77365 CF26JD 44423816 Ki > 1000 nM T77365 CE76XB 44423817 Ki > 1000 nM T77365 C5J3PM 44423818 Ki > 1000 nM T77365 CA2HW6 44423819 Ki > 1000 nM T77365 CFM1I4 44423820 Ki > 1000 nM T77365 CFTE30 44423821 Ki > 1000 nM T77365 CQL6J8 44423822 Ki > 1000 nM T77365 C4QFX3 44423823 Ki > 1000 nM T77365 CWQK67 44423824 Ki > 1000 nM T77365 CG5O9I 44423825 Ki > 1000 nM T77365 CK1EQ6 44423826 Ki > 1000 nM T77365 C4ZL9F 44423827 Ki > 1000 nM T77365 CH96WQ 44423828 Ki > 1000 nM T77365 CLJ9T4 44423837 Ki > 1000 nM T77365 CT1YQ4 44423838 Ki > 1000 nM T77365 CWL9P8 44427581 Ki = 486 nM T77365 CVA8F6 44427583 Ki = 1500 nM T77365 C7L2KY 44427585 Ki = 2680 nM T77365 C7PT2S 44430151 Ki = 1800 nM T77365 CBW73G 44430154 Ki = 2410 nM T77365 CDU4P8 44430156 Ki = 726 nM T77365 CA9L1D 44430158 Ki = 1410 nM T77365 C9M0OF 44430160 Ki > 5000 nM T77365 C0HBJ8 44430163 Ki > 4000 nM T77365 CQF30M 44430165 Ki > 5000 nM T77365 C2F3ZV 44430169 Ki > 5000 nM T77365 C4IT7U 44430170 Ki > 5000 nM T77365 C4S5DC 44430171 Ki > 5000 nM T77365 CYS8I1 44430173 Ki > 5000 nM T77365 CLW6M5 44430177 Ki > 5000 nM T77365 CZ2CX5 44430187 Ki > 5000 nM T77365 C42LMQ 44430188 Ki > 5000 nM T77365 C0UDY1 44430192 Ki > 5000 nM T77365 C87TZB 44430198 Ki = 2320 nM T77365 CI97LW 44430203 Ki > 5000 nM T77365 CPW14D 44430206 Ki = 1180 nM T77365 CNX54A 44430209 Ki = 1480 nM T77365 CC20AB 44430231 Ki = 239 nM T77365 C09MBQ 44430232 Ki = 1170 nM T77365 CDH26R 44430235 Ki = 357 nM T77365 C8UN2W 44430236 Ki > 5000 nM T77365 CX5RU6 44430239 Ki > 5000 nM T77365 CL6C1D 44430241 Ki > 5000 nM T77365 C41XMS 44435352 Ki = 9700 nM T77365 CLA42W 44435353 Ki = 5500 nM T77365 CATF75 44435354 Ki > 100000 nM T77365 CUFC32 44435355 Ki > 100000 nM T77365 C60SDL 44435356 Ki > 100000 nM T77365 CS7P6L 44435357 Ki = 7800 nM T77365 C08PCX 44435358 Ki = 34700 nM T77365 C18ANC 44435359 Ki > 100000 nM T77365 C3GB1N 44435360 Ki > 100000 nM T77365 CYP61J 44435361 Ki > 100000 nM T77365 C21UTJ 44437214 EC50 = 302 nM T77365 CAO98V 44437220 Ki = 4560 nM T77365 C67ZNA 44437460 Ki = 2030 nM T77365 CS4F7L 44438074 Ki = 6.3 nM T77365 C9BD5R 44438075 Ki = 4.1 nM T77365 CFI65U 44438076 Ki = 1.7 nM T77365 C2U6GI 44438077 Ki = 1.5 nM T77365 CIG1E4 44438078 Ki = 4.6 nM T77365 CX70ZG 44438079 Ki = 1.7 nM T77365 C0RKI1 44438080 Ki = 4.6 nM T77365 CCD9H8 44438081 Ki = 0.1 nM T77365 CWE86M 44438082 Ki = 0.4 nM T77365 CVZ37U 44438083 Ki = 0.9 nM T77365 C5DZX4 44438084 Ki = 0.3 nM T77365 CNCH68 44438085 Ki = 0.4 nM T77365 C6D3BW 44438086 Ki = 1.7 nM T77365 CD81YT 44438087 Ki = 0.9 nM T77365 CDGP07 44438088 Ki = 3.7 nM T77365 C80HQI 44438089 Ki = 2 nM T77365 C56YGL 44438090 Ki = 9.3 nM T77365 C4PL3J 44438091 Ki = 10 nM T77365 CT3P7I 44438092 Ki = 20.5 nM T77365 C4RQC0 44438093 Ki = 89.7 nM T77365 CEJ7B1 44439732 Ki = 1.3 nM T77365 C0ECH8 44439733 Ki = 1.4 nM T77365 C9OL4A 44439734 Ki = 2.1 nM T77365 CU3PC7 44439735 Ki = 0.5 nM T77365 CTLG71 44439736 Ki = 0.6 nM T77365 C7RU9N 44439737 Ki = 1.4 nM T77365 CC5KT8 44439738 Ki = 0.6 nM T77365 C04FPR 44439771 Ki = 0.6 nM T77365 CYF7C4 44439772 Ki = 1.6 nM T77365 CLM6O3 44439773 Ki = 0.8 nM T77365 CS0N7O 44439774 Ki = 2.2 nM T77365 CQ3NZ5 44439775 Ki = 0.6 nM T77365 C71WYB 44439776 Ki = 0.6 nM T77365 CYB86Z 44442015 Ki > 10000 nM T77365 C1UIO8 44442016 Ki > 10000 nM T77365 CUP5T0 44442018 Ki > 10000 nM T77365 C4RDK6 44442019 Ki > 10000 nM T77365 CPC63E 44442162 Ki > 10000 nM T77365 C71XQS 44442163 Ki > 10000 nM T77365 C42ZRD 44442166 Ki > 10000 nM T77365 C9Z3CW 44442167 Ki > 10000 nM T77365 C06RLU 44446477 Ki > 5000 nM T77365 CFPZ19 44447519 Ki = 10400 nM T77365 CJ7MS5 44447534 Ki > 100000 nM T77365 C3LOJ1 44447535 Ki = 15900 nM T77365 C95AWU 44448014 Ki = 16 nM T77365 CL3WE0 44448018 Ki = 7.5 nM T77365 C3KQS2 44448019 Ki = 7.4 nM T77365 CGYJ03 44448021 Ki = 11 nM T77365 CU02SC 44448022 Ki > 10000 nM T77365 CYD75N 44448023 Ki = 6.8 nM T77365 CTAH78 44448024 Ki = 14 nM T77365 CMJ65Z 44448025 Ki = 36 nM T77365 CHA97I 44448026 Ki = 3.7 nM T77365 CX64PJ 44448028 Ki > 10000 nM T77365 CRU9L2 44448032 Ki = 3.6 nM T77365 C9I0XB 44448036 Ki = 1.8 nM T77365 C4NM9H 44448051 Ki = 0.3 nM T77365 CQ6BZ5 44448052 Ki = 1 nM T77365 CRO52K 44448053 Ki = 1.2 nM T77365 C9FIN4 44448055 Ki = 3.7 nM T77365 CAOB06 44448056 Ki = 0.7 nM T77365 C2UWA8 44449279 Ki = 71 nM T77365 CR4Z0Q 44449308 Ki = 340 nM T77365 C8J0NG 44449493 Ki = 102 nM T77365 CV63AZ 44449494 Ki = 23 nM T77365 CKL58O 44449520 Ki = 13 nM T77365 C60TLI 44449522 Ki = 56 nM T77365 CME34Q 44449532 Ki = 2.8 nM T77365 CL4HT0 44449533 Ki = 3.6 nM T77365 C6Z1WI 44449555 Ki = 13 nM T77365 C62URD 44449567 Ki = 81 nM T77365 CO8P4M 44449568 Ki = 26 nM T77365 CO04QJ 44449570 Ki = 3079 nM T77365 C9ZH1F 44449591 Ki = 26 nM T77365 CI80QT 44449598 Ki = 299 nM T77365 C19JVY 44449599 Ki = 14 nM T77365 CZ95HM 44449626 Ki = 206 nM T77365 C9OU7X 44449633 Ki = 203 nM T77365 C0PO3H 44449634 Ki = 748 nM T77365 CZUB58 44449635 Ki = 2.3 nM T77365 C80YCR 44449636 Ki = 60 nM T77365 C0LAZ6 44449655 Ki = 779 nM T77365 CRES01 44449665 Ki = 40 nM T77365 C9ODF3 44449666 Ki = 58 nM T77365 C74VPR 44449668 Ki = 1326 nM T77365 C5X0UL 44449693 Ki = 4105 nM T77365 CXK0M2 44449706 Ki = 142 nM T77365 C1DLR5 44449707 Ki = 779 nM T77365 C0HZ1F 44449728 Ki = 45 nM T77365 CLGN80 44449740 Ki = 172 nM T77365 C6SMZ7 44449742 Ki = 55 nM T77365 C9KA4M 44449744 Ki = 444 nM T77365 C95SAB 44449745 Ki = 154 nM T77365 C3N9OC 44449746 Ki = 6493 nM T77365 CP78RA 44450158 Ki = 30 nM T77365 C0E3MF 44450161 Ki = 33 nM T77365 C6I3MS 44450188 Ki = 5737 nM T77365 C0SU7H 44450189 Ki = 435 nM T77365 C8W5YK 44450190 Ki = 1384 nM T77365 CHP5W0 44450290 Ki = 1.8 nM T77365 C5EFV0 44450384 Ki = 3.8 nM T77365 CCMZ32 44450517 Ki = 181 nM T77365 C6Y0PD 44450826 Ki = 239.88 nM T77365 C6J4IM 44450828 Ki = 208.93 nM T77365 C6VFH5 44450829 Ki = 426.58 nM T77365 C7UPI4 44450849 Ki = 158.49 nM T77365 CSO5T9 44450850 Ki = 74.13 nM T77365 CR79ZP 44450903 Ki = 870.96 nM T77365 CR5BE0 44450904 Ki = 588.84 nM T77365 CU4SW3 44450905 Ki = 1047.13 nM T77365 CN38SJ 44450929 Ki = 1148.15 nM T77365 CTBV26 44450930 Ki = 302 nM T77365 CHU69T 44450931 Ki = 794.33 nM T77365 CJ6D7U 44450932 Ki = 38.02 nM T77365 CA01KF 44450933 Ki = 239.88 nM T77365 CGXZ65 44450955 Ki = 398.11 nM T77365 CQ6K2P 44450979 Ki = 407.38 nM T77365 C8XGN7 44450981 Ki = 323.59 nM T77365 C76MCE 44450982 Ki = 3548.13 nM T77365 C6PK0V 44450983 Ki = 257 nM T77365 CVC48J 44450997 Ki = 1023.29 nM T77365 CGW63R 44451018 Ki = 223.87 nM T77365 C76WNY 44451019 Ki = 707.95 nM T77365 CCF1X3 44451020 Ki = 691.83 nM T77365 C5J8RO 44451021 Ki = 162.18 nM T77365 CEN6T1 44451048 Ki = 467.74 nM T77365 CSH7C2 44451049 Ki = 1096.48 nM T77365 C0N8UL 44451050 Ki = 316.23 nM T77365 C1J9DN 44451053 Ki = 173.78 nM T77365 C3F9IW 44451073 Ki = 48.98 nM T77365 C1Z9JQ 44451074 Ki = 478.63 nM T77365 CASC19 44451075 Ki = 114.82 nM T77365 CL4H9C 44451099 Ki = 398.11 nM T77365 CN4GU2 44451100 Ki = 630.96 nM T77365 CV4I0S 44451106 Ki = 794.33 nM T77365 C4N3OQ 44451123 Ki = 645.65 nM T77365 CNEP36 44451126 Ki = 562.34 nM T77365 CN7TA8 44451127 Ki = 323.59 nM T77365 C6JO2N 44451128 Ki = 741.31 nM T77365 CHZU82 44451129 Ki = 707.95 nM T77365 CZB19U 44451169 Ki = 1445.44 nM T77365 CPGH68 44451171 Ki = 1548.82 nM T77365 CPX20Z 44451197 Ki = 6760.83 nM T77365 CXYO54 44451199 Ki = 263.03 nM T77365 CKM13P 44451200 Ki = 151.36 nM T77365 CKIL97 44451201 Ki = 1584.89 nM T77365 C75LZM 44451224 Ki = 12022.64 nM T77365 CPL9E7 44451229 Ki = 812.83 nM T77365 C52UIJ 44451230 Ki = 154.88 nM T77365 CJEA96 44451252 Ki = 169.82 nM T77365 C8CQ3K 44451253 Ki = 323.59 nM T77365 C2Y9WZ 44451254 Ki = 10000 nM T77365 CMN2L6 44451269 Ki = 269.15 nM T77365 CUE61I 44451271 Ki = 323.59 nM T77365 C7HMX9 44451272 Ki = 354.81 nM T77365 C50QVJ 44451283 Ki = 107.15 nM T77365 CUA67B 44451284 Ki = 354.81 nM T77365 C74QDH 44451285 Ki = 131.83 nM T77365 C3OM0Y 44451303 Ki = 181.97 nM T77365 CAL31F 44451305 Ki = 114.82 nM T77365 CJO78N 44451306 Ki = 398.11 nM T77365 C9U8GO 44451329 Ki = 389.05 nM T77365 C21QUX 44451330 Ki = 154.88 nM T77365 CMQ4H8 44451480 Ki = 2344.23 nM T77365 CEL5J8 44451482 Ki = 7079.46 nM T77365 C0ZD4U 44451483 Ki = 173.78 nM T77365 C0TLS7 44451489 Ki = 616.6 nM T77365 CEG1Y5 44451491 Ki = 416.87 nM T77365 CE9Q5B 44451492 Ki = 354.81 nM T77365 CYOF07 44451499 Ki = 69.2 nM T77365 CO0UD1 44451500 Ki = 222 nM T77365 CGS85Y 44451501 Ki = 574 nM T77365 CL8PQ6 44451524 Ki = 339 nM T77365 C3VZR4 44451525 Ki = 54.5 nM T77365 C1T8VP 44451582 Ki = 48.2 nM T77365 C8JOS1 44451604 Ki = 557 nM T77365 CN7KU2 44451658 Ki = 158 nM T77365 CG1FV5 44451682 Ki = 300 nM T77365 C0JB2Q 44451683 Ki = 21.3 nM T77365 C4J3XI 44451738 Ki = 27.2 nM T77365 C8GL3J 44451787 Ki = 49.8 nM T77365 C8M6EA 44451790 Ki = 5.2 nM T77365 COVW35 44451815 Ki = 69.5 nM T77365 C3UIY5 44451817 Ki = 32.9 nM T77365 CA76ZH 44451846 Ki = 280 nM T77365 C1DVS2 44451849 Ki = 45.5 nM T77365 CDP23H 44451903 Ki = 35.3 nM T77365 CN0BP8 44452405 Ki = 302 nM T77365 C4APQ6 44452407 Ki = 64.57 nM T77365 C1KXG7 44452431 Ki = 398.11 nM T77365 C6AG2Y 44452434 Ki = 158.49 nM T77365 CJW91V 44452435 Ki = 63.1 nM T77365 C87QHW 44452454 Ki = 575.44 nM T77365 C0PER5 44452455 Ki = 199.53 nM T77365 C3G5HY 44452478 Ki = 398.11 nM T77365 CTC57Y 44452490 Ki = 109.65 nM T77365 CBM43V 44452492 Ki = 309.03 nM T77365 CTMF29 44452493 Ki = 398.11 nM T77365 C6DU3Q 44452514 Ki = 371.54 nM T77365 CG74SF 44452515 Ki = 3090.3 nM T77365 C18BXC 44452535 Ki = 63.1 nM T77365 CWF9E6 44452536 Ki = 47.86 nM T77365 CSFV93 44452539 Ki = 51.29 nM T77365 C8SIX2 44452695 Ki = 489.78 nM T77365 CQ7RM8 44454227 IC50 = 60 nM T77365 CKE80T 44454230 IC50 = 1000 nM T77365 CDL69J 44454231 IC50 = 1010 nM T77365 C91PTR 44454502 Ki = 6 nM T77365 CCX38P 44454534 Ki = 10 nM T77365 C5S4NW 44454568 Ki = 0.8 nM T77365 C7ZF2J 44454569 Ki = 0.2 nM T77365 C7W3MH 44454595 Ki = 2 nM T77365 CL4GC7 44454626 Ki = 5 nM T77365 C5MGR8 44454628 Ki = 3 nM T77365 CD3HE5 44454670 Ki = 3 nM T77365 CJ6N1L 44454671 Ki = 1 nM T77365 C9M3PR 44454697 Ki = 1 nM T77365 C75VEK 44454726 Ki = 3 nM T77365 C4B7VM 44454763 IC50 >= 10000 nM T77365 C2EQM1 44454764 IC50 >= 10000 nM T77365 CO3BX7 44454781 Ki = 5 nM T77365 CWZG75 44454788 IC50 >= 10000 nM T77365 C9YD4Q 44454789 IC50 >= 10000 nM T77365 CK37UL 44454808 Ki = 5 nM T77365 CN7Y2F 44454816 IC50 >= 10000 nM T77365 CTWR48 44454817 IC50 >= 10000 nM T77365 CU5XL2 44454818 IC50 >= 10000 nM T77365 CL6KS1 44454834 Ki = 2 nM T77365 C8UI0N 44454836 Ki = 2 nM T77365 CB67EY 44454849 IC50 >= 10000 nM T77365 C60CIT 44454850 IC50 >= 10000 nM T77365 CZU8C6 44454851 IC50 >= 10000 nM T77365 CH5SW9 44454853 IC50 >= 10000 nM T77365 CL39AN 44454883 IC50 >= 10000 nM T77365 C7UK9H 44454885 IC50 >= 10000 nM T77365 C52HBA 44454886 IC50 >= 10000 nM T77365 C0ET4C 44454907 Ki = 4 nM T77365 C7APO0 44454922 IC50 >= 10000 nM T77365 C52LGN 44454923 IC50 >= 10000 nM T77365 C6CO9J 44454925 IC50 >= 10000 nM T77365 CHY9A8 44454940 Ki = 1 nM T77365 C6L0ZS 44454941 Ki = 1 nM T77365 C9JL7N 44457461 Ki = 4190 nM T77365 CXOS03 44457466 Ki = 6940 nM T77365 C6A9OT 44457469 Ki = 10100 nM T77365 CS1F5E 44457473 Ki = 893 nM T77365 CR58PU 44457922 Ki = 59 nM T77365 CIDT05 44457923 Ki = 5.48 nM T77365 C0GTF5 44457953 Ki = 120 nM T77365 C2GTV4 44458220 Ki = 6 nM T77365 CQ0WM7 44469273 IC50 > 5000 nM T77365 C4DL5C 44469677 IC50 > 10000 nM T77365 C2T8CA 44520931 Ki = 4.9 nM T77365 CT8OY0 44520932 Ki = 12.3 nM T77365 CXU2F8 44520933 Ki = 7.5 nM T77365 C5V6OI 44520934 Ki = 6.5 nM T77365 CKC3Q4 44520935 Ki = 25 nM T77365 C6H7PM 44520936 Ki = 88 nM T77365 CLCB53 44520937 Ki = 420 nM T77365 CD29LZ 44520938 Ki = 18.6 nM T77365 CI82SB 44520939 Ki = 8.8 nM T77365 CC97FL 44520940 Ki = 126 nM T77365 CB7K2Y 44520941 Ki = 4 nM T77365 CL3NH5 44520942 Ki = 14 nM T77365 CU3GW7 44520943 Ki = 17 nM T77365 C6CEV4 44520944 Ki = 18 nM T77365 CD9Q7Z 44520945 Ki = 31 nM T77365 CCS87V 44520946 Ki = 31 nM T77365 C21CFR 44520947 Ki = 49 nM T77365 C6HN5S 44520948 Ki = 18 nM T77365 C8DZR0 44520949 Ki = 36 nM T77365 CH7FI4 44520950 Ki = 57 nM T77365 CO82QN 44520951 Ki = 28 nM T77365 CGH3X0 44520952 Ki = 153 nM T77365 CJ4NA8 44520953 Ki = 92 nM T77365 C49KZA 44520954 Ki = 253 nM T77365 CW76RP 44520955 Ki = 255 nM T77365 CQK20C 44520956 Ki = 3290 nM T77365 C6KJC7 44520957 Ki = 14 nM T77365 CIR5M0 44520958 Ki = 9 nM T77365 CMU48O 44520959 Ki = 24 nM T77365 C5L2GJ 44520960 Ki = 23 nM T77365 CN0MR1 44520961 Ki = 9 nM T77365 C7AGL5 44520962 Ki = 16 nM T77365 CWV6A8 44520963 Ki = 30 nM T77365 CWR28D 44520964 Ki = 24 nM T77365 C9HO8N 44520965 Ki = 155 nM T77365 C4RDH8 44520966 Ki = 107 nM T77365 C38PAD 44520967 Ki = 107 nM T77365 C5QPO3 44520968 Ki = 123 nM T77365 CZ4I9A 44520969 Ki = 29 nM T77365 C8Y4MD 44520970 Ki = 2450 nM T77365 CZ37SW 44520971 Ki = 12 nM T77365 CZO52W 44520972 Ki = 25 nM T77365 CK69IO 44520973 Ki = 155 nM T77365 CEP2L4 44520974 Ki = 183 nM T77365 CJ97HI 44520975 Ki = 97 nM T77365 CZ6F9S 44520976 Ki = 2.5 nM T77365 C4Q5JZ 44520977 Ki = 3 nM T77365 CX54QG 44520978 Ki = 9.5 nM T77365 C9EH4F 44520979 Ki = 3 nM T77365 CQ71XC 44520980 Ki = 2.5 nM T77365 CEO4P7 44520981 Ki = 2 nM T77365 C31SUP 44520982 Ki = 1 nM T77365 CNR53B 44520983 Ki = 3.5 nM T77365 C3ZCH7 44520984 Ki = 6 nM T77365 C3MZC5 44520985 Ki = 5.5 nM T77365 C7HVU4 44520987 Ki = 3 nM T77365 C5M3GT 44520988 Ki = 6 nM T77365 CJ57RW 44537897 Ki = 5.43 nM T77365 C9SK6P 44551168 Ki = 83.18 nM T77365 C9O6XK 44560456 Ki = 4.1 nM T77365 C85JWE 44560507 Ki = 1.5 nM T77365 CVW3N2 44563977 Ki = 2100 nM T77365 C4LI1U 44564568 Ki = 111 nM T77365 C4VJB3 44564569 Ki = 261 nM T77365 CJ94UT 44564881 Ki = 24 nM T77365 CVUD54 44564882 Ki = 1561 nM T77365 C75ZAH 44564883 Ki = 409 nM T77365 CI9BH4 44564926 Ki = 89 nM T77365 CPF51G 44564927 Ki = 316 nM T77365 CD0W8R 44564928 Ki = 2587 nM T77365 CUX0Q7 44564978 Ki = 9213 nM T77365 CL72ZU 44564979 Ki = 54 nM T77365 CP2FL0 44564980 Ki = 33 nM T77365 CO1Z3J 44564981 Ki = 86 nM T77365 CIEH58 44565032 Ki = 6 nM T77365 CFJ49P 44565033 Ki = 359 nM T77365 CJ9T8U 44565034 Ki = 2641 nM T77365 CTYJ67 44565076 Ki = 5122 nM T77365 C9WV1X 44565077 Ki = 23 nM T77365 C65ZWP 44565078 Ki = 31 nM T77365 CO1RK2 44565079 Ki = 60 nM T77365 C5C3RG 44565133 Ki = 72 nM T77365 CA5B6M 44565134 Ki = 106 nM T77365 CFJ6D2 44565135 Ki = 213 nM T77365 C1LK8I 44565136 Ki = 499 nM T77365 C2B3MD 44565183 Ki = 12 nM T77365 C6TXF8 44565184 Ki = 50 nM T77365 CV6I0P 44567439 Ki = 80600 nM T77365 CT51OW 44568290 Ki = 1.1 nM T77365 C8PZ3K 44568291 Ki = 0.5 nM T77365 CG7N0U 44568314 Ki = 7.8 nM T77365 CN3F0X 44568315 Ki = 1.9 nM T77365 CXA9V7 44568316 Ki = 0.6 nM T77365 C9R2WY 44568344 Ki = 5.5 nM T77365 C3ZOE0 44568345 Ki = 11.4 nM T77365 CCN6H0 44568373 Ki = 2.7 nM T77365 C9FXY3 44568374 Ki = 2.8 nM T77365 C6GNF2 44568375 Ki = 1.5 nM T77365 CNK5F8 44568376 Ki = 2.3 nM T77365 CT1DS3 44568401 Ki = 1.6 nM T77365 CR48BE 44568402 Ki = 1.3 nM T77365 C3H9EA 44568403 Ki = 1.8 nM T77365 C2RJ7Q 44568838 Ki = 475 nM T77365 CW0B5D 44570367 Ki > 1000 nM T77365 C9BA3H 44570369 Ki > 1000 nM T77365 C24CRG 44570413 Ki > 1000 nM T77365 C6EAT9 44570414 Ki > 1000 nM T77365 CTS6P4 44570415 Ki > 1000 nM T77365 CP93SE 44570416 Ki > 1000 nM T77365 C6NJP3 44570454 Ki > 1000 nM T77365 CC6TW2 44570455 Ki > 1000 nM T77365 CG9BR2 44570456 Ki > 1000 nM T77365 C9FV0G 44570457 Ki > 1000 nM T77365 CC51RV 44570458 Ki > 1000 nM T77365 CSMN18 44570493 Ki > 1000 nM T77365 C5KUC7 44571407 Ki = 1 nM T77365 C1ZQ2Y 44571408 Ki = 1.8 nM T77365 CJEC97 44571505 Ki = 46 nM T77365 CJI0N2 44571506 Ki = 5.7 nM T77365 CHK25M 44571507 Ki = 2 nM T77365 CEV3M2 44571508 Ki = 3 nM T77365 CM8Y1O 44571550 Ki = 6 nM T77365 CZ16AK 44571551 Ki = 2.8 nM T77365 CF09TO 44571585 Ki = 9.5 nM T77365 CUFW23 44571671 Ki = 1.5 nM T77365 CDQ4I2 44571672 Ki = 0.7 nM T77365 CMY36G 44571722 Ki = 0.8 nM T77365 CU63ZL 44571767 Ki = 0.3 nM T77365 CR8B1D 44571835 Ki = 0.3 nM T77365 CMD87Q 44572294 Ki > 100000 nM T77365 CSL0G8 44572353 Ki > 100000 nM T77365 C0ETQ1 44572354 Ki > 100000 nM T77365 C7D2GC 44572410 Ki > 100000 nM T77365 C9VS8P 44572470 Ki > 100000 nM T77365 CDZ14G 44572472 Ki > 100000 nM T77365 C8Y0EI 44574117 Ki = 34.7 nM T77365 CZDG39 44574118 Ki = 72.4 nM T77365 CZX7N5 44574165 Ki = 10.5 nM T77365 C6TIR8 44574166 Ki = 15.1 nM T77365 CLTE07 44574167 Ki = 490 nM T77365 CJ3LA8 44574168 Ki = 18.2 nM T77365 CWDA90 44574191 Ki = 132 nM T77365 C0BP3Z 44574192 Ki = 43.7 nM T77365 CX6KL4 44574193 Ki = 1000 nM T77365 CUH78B 44574194 Ki = 28.8 nM T77365 CMFB42 44574222 Ki = 118 nM T77365 C4VBL3 44574223 Ki = 3311 nM T77365 CSA38M 44574224 Ki = 2240 nM T77365 CUBQ21 44574225 Ki = 35.5 nM T77365 CY14AD 44574251 Ki = 21.9 nM T77365 C7GY5T 44574252 Ki = 10 nM T77365 CPH71S 44574253 Ki = 447 nM T77365 C4V5GO 44574254 Ki = 28.2 nM T77365 CN2OG0 44574281 Ki = 50.1 nM T77365 C8BZ5U 44577872 Ki = 4 nM T77365 CA31JY 44579667 Ki = 4770 nM T77365 CR0GX1 44579668 Ki = 1670 nM T77365 CF04WK 44579673 Ki = 2620 nM T77365 CRS81G 44579674 Ki = 6870 nM T77365 CF2O3K 44579675 Ki = 2010 nM T77365 CL18FO 44579714 Ki = 1080 nM T77365 C5TKU6 44579715 Ki = 4510 nM T77365 CI4FW1 44579716 Ki = 1600 nM T77365 CZ7NV2 44579717 Ki = 1530 nM T77365 CHC02W 44581364 Ki = 67 nM T77365 C0X4UM 44581365 Ki = 89 nM T77365 CHR9Z1 44581366 Ki = 195 nM T77365 CB1Q8U 44581367 Ki = 154 nM T77365 CINU98 44581368 Ki = 281 nM T77365 CMB71E 44581369 Ki = 455 nM T77365 C27QRK 44581397 Ki = 105 nM T77365 CS8QR0 44581398 Ki = 61 nM T77365 C9S3YK 44581428 Ki = 12 nM T77365 CDT8Z2 44581429 Ki = 105 nM T77365 CWBF57 44581430 Ki = 6818 nM T77365 C8ZU0M 44581431 Ki = 2798 nM T77365 C60UGT 44581432 Ki = 160 nM T77365 C7CAH0 44581471 Ki = 8170 nM T77365 C76WPB 44581472 Ki = 7140 nM T77365 CZ72WU 44581866 Ki = 26 nM T77365 C8FEZ9 44581894 Ki = 25.8 nM T77365 CM6AK4 44581895 Ki = 275 nM T77365 C6EUC0 44581896 Ki = 47 nM T77365 CCB34Q 44582614 Ki = 2050 nM T77365 CSM58E 44582652 Ki = 24000 nM T77365 CA5R4M 44582653 Ki = 31600 nM T77365 CR95SV 44582654 Ki = 5170 nM T77365 C8G4TH 44582690 Ki > 100000 nM T77365 CV5F9X 44582691 Ki > 100000 nM T77365 C71SDJ 44582723 Ki = 18900 nM T77365 CLW60K 44582724 Ki = 8780 nM T77365 CH07JS 44582725 Ki = 11800 nM T77365 CZ91EO 44582726 Ki = 797 nM T77365 CR3LW0 44583035 Ki = 10000 nM T77365 CY2MH0 44586253 Ki = 158.3 nM T77365 CC7FH5 44586717 Ki = 397 nM T77365 C7S1MY 44586718 Ki = 188 nM T77365 CLZ6A1 44587954 Ki = 933 nM T77365 C6B4KH 44587955 Ki = 408 nM T77365 C6IO7C 44587956 Ki = 100 nM T77365 CUG8E4 44587957 Ki = 92 nM T77365 C3FQ9A 44588393 Ki = 692 nM T77365 CG1JD0 44588395 Ki = 50 nM T77365 CV6LB9 44588396 Ki = 398 nM T77365 CNG85D 44588436 Ki = 89 nM T77365 C36UPO 44588437 Ki = 240 nM T77365 C71HQU 44588438 Ki = 166 nM T77365 CD97HM 44588439 Ki = 48 nM T77365 CX7YZ2 44588470 Ki = 102 nM T77365 C5QB8V 44588471 Ki = 118 nM T77365 CWN0S7 44588472 Ki = 199 nM T77365 C4JS6Y 44588473 Ki = 631 nM T77365 C4UT7D 44588474 Ki = 148 nM T77365 CN8Q2U 44588514 Ki = 324 nM T77365 CN0M8J 44588515 Ki = 145 nM T77365 CBL10K 44588516 Ki = 28 nM T77365 C0UD5O 44588517 Ki = 468 nM T77365 C83AJU 44588518 Ki = 104 nM T77365 CZV5Q3 44589759 Ki = 2 nM T77365 C6W2RF 44589796 Ki = 17 nM T77365 CLJO67 44589797 Ki = 7 nM T77365 CMS0Z3 44589798 Ki = 2 nM T77365 C8BQJ5 44589799 Ki = 2 nM T77365 C0X8MI 44589833 Ki = 2 nM T77365 CP1M4S 44589834 Ki = 8 nM T77365 CUT65Z 44589835 Ki = 19 nM T77365 CFS08D 44589836 Ki = 2 nM T77365 CT3A1B 44589887 Ki = 4 nM T77365 CF1H2T 44589888 Ki = 3 nM T77365 CB2Z9T 44589889 Ki = 2 nM T77365 CNZQ14 44589890 Ki = 5 nM T77365 C7ZSA5 44589891 Ki = 2 nM T77365 C3PO2I 44589942 Ki = 3 nM T77365 CW76ND 44589943 Ki = 3 nM T77365 C6G7EC 44589944 Ki = 6 nM T77365 CQ4YE7 44589945 Ki = 1 nM T77365 C9K6TB 44589994 Ki = 4 nM T77365 CT3YK0 44589995 Ki = 2 nM T77365 CU3B4T 44589996 Ki = 67 nM T77365 CWV64B 44589997 Ki = 73 nM T77365 CT4F5O 44590096 Ki = 1 nM T77365 C59MHC 44590097 Ki = 2 nM T77365 C0D8HM 44590292 Ki = 297 nM T77365 CB9JU6 44590773 Ki = 110 nM T77365 CJT42W 44590830 Ki = 119 nM T77365 CWM48B 44590832 Ki = 305 nM T77365 CX98IZ 44590914 Ki = 573 nM T77365 CDJ76M 44590915 Ki = 161 nM T77365 CZL3S9 44597752 Ki = 4730 nM T77365 CVW37M 44597868 Ki = 4520 nM T77365 CV4TA7 44597869 Ki = 4520 nM T77365 C5KTS9 44597870 Ki = 4000 nM T77365 CUO03D 44597871 Ki = 1640 nM T77365 CM43HO 44598050 Ki = 372 nM T77365 C5ZLC3 44598835 Ki = 12700 nM T77365 C6LXZ8 44598836 Ki = 24300 nM T77365 CFIA83 44631910 IC50 > 50000 nM T77365 CK05TD 45106502 Ki = 2511.89 nM T77365 CDTA58 45136848 Ki = 6.2 nM T77365 C36SXK 45136852 Ki = 6.5 nM T77365 CLB20G 45266415 Ki > 100000 nM T77365 CU84YS 45266426 Ki > 100000 nM T77365 CNO3D6 45267119 Ki = 153 nM T77365 C1I6ZN 45267125 Ki = 20 nM T77365 C6BDH1 45267130 Ki = 79 nM T77365 CHK6Z9 45267243 Ki = 1400 nM T77365 CJZ29E 45267454 Ki = 3630 nM T77365 C24KLI 45267987 Ki = 7.6 nM T77365 CG7M5U 45267990 Ki = 2.6 nM T77365 C35COL 45267991 Ki = 213.8 nM T77365 C5ZFY1 45268103 Ki = 3410 nM T77365 CSGE26 45268313 Ki = 1470 nM T77365 CSP4L8 45268863 Ki = 16 nM T77365 C7T3HW 45268867 Ki = 147.91 nM T77365 C1IL3E 45268869 Ki = 3.7 nM T77365 C9WOM0 45268873 Ki = 229.09 nM T77365 CXI20R 45268920 Ki = 218.78 nM T77365 C8AL4S 45268921 Ki = 208.93 nM T77365 C5I0MX 45268927 Ki = 338.84 nM T77365 C8IM6P 45268928 Ki = 398.11 nM T77365 C7EL9J 45269703 Ki = 23 nM T77365 CU2D9I 45269706 Ki = 95.5 nM T77365 C1YSN9 45269707 Ki = 87.1 nM T77365 CW3QL8 45269711 Ki = 416.87 nM T77365 C5QT0W 45269769 Ki = 524.81 nM T77365 C57YDT 45269835 Ki = 997 nM T77365 C0Q7RF 45269838 Ki = 3630 nM T77365 CW8U6A 45270537 Ki = 170 nM T77365 CJP69G 45270541 Ki = 4.8 nM T77365 C5HQ6O 45270544 Ki = 204.17 nM T77365 CX78GF 45271359 Ki = 308 nM T77365 CTL27N 45271361 Ki = 56.23 nM T77365 CK52VZ 45271363 Ki = 758.58 nM T77365 CY3A1D 45271366 Ki = 17.5 nM T77365 C20RJQ 45271709 Ki = 570 nM T77365 CK1H3O 45272255 Ki = 220 nM T77365 CZ3D2A 45272256 Ki = 10 nM T77365 CNAT29 45272259 Ki = 169.82 nM T77365 CQ6N7W 45272308 Ki = 489.78 nM T77365 C48IEM 45272391 Ki = 6560 nM T77365 C5YT4Z 45273099 Ki = 5011.87 nM T77365 CS4L5G 45273118 Ki = 1778.28 nM T77365 C6O8XQ 45273122 Ki = 9.5 nM T77365 C5SRP3 45274224 Ki = 26 nM T77365 CAM9S8 45274225 Ki = 17.1 nM T77365 CWZV56 45274227 Ki = 168 nM T77365 C9MB3Z 45274228 Ki = 57 nM T77365 C19YWV 45274324 Ki = 2.4 nM T77365 CV4R3I 45274328 Ki = 6.9 nM T77365 C5OBS2 45274330 Ki = 2.9 nM T77365 CU4XV8 45274426 Ki = 13.1 nM T77365 CS3CF1 45274431 Ki = 25.2 nM T77365 CBX3M6 45275056 Ki = 11.4 nM T77365 CBUV31 45275058 Ki = 29.8 nM T77365 C6TC5O 45275060 Ki = 63.4 nM T77365 CE7F8G 45275061 Ki = 222 nM T77365 CS86LV 45275168 Ki > 1000 nM T77365 CSEL27 45275170 Ki = 340 nM T77365 CYL7Z2 45275171 Ki = 1016 nM T77365 CUMC92 45275172 Ki = 118 nM T77365 CV7L4T 45275173 Ki = 42 nM T77365 C8LB2S 45275287 Ki = 1.4 nM T77365 COVY03 45275517 Ki = 11.1 nM T77365 CX49ZH 45275619 Ki = 49 nM T77365 CCL28P 45275713 Ki = 107 nM T77365 CK2G4Y 45275714 Ki = 31 nM T77365 C4ZT2C 45275715 Ki = 11 nM T77365 CTN65H 45275716 Ki = 215 nM T77365 CP82KG 45275717 Ki = 16.1 nM T77365 CQC5T8 45275718 Ki = 13.2 nM T77365 CU8HY4 45275719 Ki = 40.1 nM T77365 CLE92Q 45275818 Ki = 100 nM T77365 C8P0ZA 45275819 Ki = 304 nM T77365 CQL3P8 45275820 Ki = 539 nM T77365 C6BIV9 45275821 Ki = 9 nM T77365 CX5F0H 45275823 Ki = 203 nM T77365 C8DPZ0 45275824 Ki = 263 nM T77365 CO2E5P 45278533 Ki = 6.6 nM T77365 C3WGV4 45278535 Ki = 350 nM T77365 CJED13 45278537 Ki = 110 nM T77365 CC4XE8 45278538 Ki = 39 nM T77365 CIV2G3 45278539 Ki = 180 nM T77365 CQYO92 45278617 Ki = 83.5 nM T77365 C1GP7V 45278618 Ki > 10000 nM T77365 C6WVU9 45278619 Ki = 390 nM T77365 CNG16P 45278621 Ki = 13.2 nM T77365 CQ5J7L 45278622 Ki = 238 nM T77365 C15LZX 45278623 Ki = 240 nM T77365 C93ZXP 45278697 Ki = 300 nM T77365 CHL5W1 45278699 Ki = 1030 nM T77365 C9V6XY 45278700 Ki = 36.1 nM T77365 CMJ06I 45278701 Ki = 360 nM T77365 CD7GE2 45278783 Ki = 54.4 nM T77365 CVDZ38 45278784 Ki = 50.9 nM T77365 CUE83H 45278785 Ki = 370 nM T77365 CVDJ21 45278787 Ki = 97.7 nM T77365 CXU4S7 45278863 Ki = 79.2 nM T77365 CKVQ57 45278864 Ki = 36.7 nM T77365 CG23WV 45278865 Ki = 22.2 nM T77365 CZI7V5 45278866 Ki = 33.4 nM T77365 CJ5G3X 45278867 Ki = 8.7 nM T77365 CJ1MA9 45278868 Ki = 11 nM T77365 CX4B6U 45278944 Ki = 10 nM T77365 C5S6IP 45278946 Ki = 42.2 nM T77365 C3LI4D 45278947 Ki = 43.2 nM T77365 CZ7T1U 45278948 Ki = 28.6 nM T77365 C96HNR 45278949 Ki = 30.8 nM T77365 CIC9V4 45279186 Ki = 9.1 nM T77365 CZ42MB 45279272 Ki = 45.4 nM T77365 CG6N9M 45279273 Ki = 15.9 nM T77365 C85DGX 45279274 Ki = 30 nM T77365 CXZ01P 45279275 Ki = 78.9 nM T77365 CJB9L4 45279276 Ki = 89.1 nM T77365 CV29MU 45279277 Ki = 17 nM T77365 CES35K 45279356 Ki = 25.2 nM T77365 C45JDQ 45279358 Ki = 210 nM T77365 CT4LX5 45279360 Ki = 1010 nM T77365 C9PV1L 45279361 Ki = 150 nM T77365 CQ7U1I 45279362 Ki = 130 nM T77365 CJL90G 45279445 Ki = 12.1 nM T77365 CU6P4F 45279446 Ki > 1360 nM T77365 CQ4WL3 45279448 Ki = 960 nM T77365 CR73ZU 45279449 Ki = 64.6 nM T77365 CMH6F3 45279451 Ki = 250 nM T77365 C64KIA 45279539 Ki = 125 nM T77365 CIZS47 45279541 Ki = 28.1 nM T77365 CJ53BU 45279542 Ki = 36 nM T77365 CN8TV0 45279543 Ki = 110 nM T77365 C1O0IT 45279544 Ki = 55.5 nM T77365 CP47WG 45279545 Ki = 170 nM T77365 C0C1LT 45279632 Ki = 28.8 nM T77365 CR07AK 45279633 Ki = 22.5 nM T77365 C15ZWH 45279636 Ki = 32.8 nM T77365 CQCA71 45279637 Ki = 26.1 nM T77365 CLEA65 45279724 Ki = 200 nM T77365 C6S0WZ 45279725 Ki = 29 nM T77365 C1H4CQ 45279727 Ki = 5.3 nM T77365 CP74GQ 45279728 Ki = 230 nM T77365 CY8R1U 45279729 Ki = 140 nM T77365 C6ZLX7 45279730 Ki = 350 nM T77365 C6MR2P 45279822 Ki = 120 nM T77365 CH52XG 45279823 Ki = 360 nM T77365 C86KCE 45279824 Ki = 10.3 nM T77365 CFV13P 45279825 Ki = 300 nM T77365 C5B7LP 45279828 Ki = 49.6 nM T77365 CO4FS7 45353990 Ki > 100000 nM T77365 CPG3L9 45481619 Ki = 1.86 nM T77365 CV13SH 45481620 Ki = 348 nM T77365 C2ZI4P 45481621 Ki = 114 nM T77365 CK2YO1 45481748 Ki = 176 nM T77365 CCMX92 45481749 Ki = 18.4 nM T77365 CXM9F4 45481750 Ki = 216 nM T77365 CBOG84 45481751 Ki = 193 nM T77365 CLZV08 45481752 Ki = 159 nM T77365 C3MPR1 45481753 Ki = 30.5 nM T77365 CB52VK 45481754 Ki = 46.5 nM T77365 C5W4NR 45481755 Ki = 8.8 nM T77365 CQOB79 45481756 Ki = 23 nM T77365 CB8NA2 45481757 Ki = 15.9 nM T77365 CL68UB 45481758 Ki = 31.3 nM T77365 CY2WO6 45481759 Ki = 9.18 nM T77365 CV43FT 45481760 Ki = 53.1 nM T77365 C50HVN 45481761 Ki = 46.9 nM T77365 C4C0QV 45481762 Ki = 52.5 nM T77365 C16LEJ 45481763 Ki = 156 nM T77365 C1TB7C 45481764 Ki = 12.9 nM T77365 CP02LD 45481765 Ki = 74.6 nM T77365 C0L9GH 45481766 Ki = 70.9 nM T77365 CH54CA 45481767 Ki = 62.5 nM T77365 C7GF4H 45481768 Ki = 15.7 nM T77365 C1FA8U 45481769 Ki = 77.5 nM T77365 C2TWL7 45481770 Ki = 42.1 nM T77365 C5H7SZ 45481771 Ki = 39.6 nM T77365 CE80TZ 45482062 Ki = 2030 nM T77365 CJG6E4 45482063 Ki = 16.1 nM T77365 CVH1A9 45482064 Ki = 3600 nM T77365 CGDC50 45482065 Ki = 3260 nM T77365 CLRE36 45482066 Ki = 31.7 nM T77365 CC3V0B 45482067 Ki = 131 nM T77365 C78IES 45482068 Ki = 2.03 nM T77365 CO96QB 45482069 Ki = 3.88 nM T77365 CDA2V1 45482070 Ki = 7.94 nM T77365 CQN78H 45482071 Ki = 15.1 nM T77365 CF9YU6 45482072 Ki = 1.95 nM T77365 C9FXY5 45482073 Ki = 8.93 nM T77365 C12JUY 45482074 Ki = 182 nM T77365 C0FG6J 45482075 Ki = 38.7 nM T77365 CQ5ZF6 45482076 Ki = 54.1 nM T77365 CMI3P8 45482077 Ki = 211 nM T77365 CDSG82 45482078 Ki = 326 nM T77365 C01FXN 45482079 Ki = 89.9 nM T77365 CE3TD2 45482080 Ki = 7.99 nM T77365 C0IT6Y 45482081 Ki = 18.7 nM T77365 C0RN6K 45482082 Ki = 11.7 nM T77365 CD6I4G 45482083 Ki = 75.9 nM T77365 CZ30JX 45482084 Ki = 73.6 nM T77365 CY49LO 45482085 Ki = 4.15 nM T77365 C1VEW8 45482086 Ki = 3.13 nM T77365 C8Q6KD 45482087 Ki = 45.2 nM T77365 CP5LN6 45482088 Ki = 39.3 nM T77365 C12UZF 45482089 Ki = 27.2 nM T77365 CIF06H 45482090 Ki = 2.75 nM T77365 CDK76E 45482091 Ki = 186 nM T77365 CC52GU 45482092 Ki = 256 nM T77365 CL39ZH 45482093 Ki = 80.5 nM T77365 C8PQ9W 45482094 Ki = 5.75 nM T77365 COL2R3 45482462 Ki = 56 nM T77365 CNDA49 45482464 Ki = 3.69 nM T77365 CLZM60 45482470 Ki = 4 nM T77365 CS1L8N 45482471 Ki = 0.43 nM T77365 CPX3O6 45482472 Ki = 75 nM T77365 CZ89HK 45482473 Ki = 5.48 nM T77365 CHV46U 45482474 Ki = 59 nM T77365 C14WOG 45482475 Ki = 50 nM T77365 CS2D7I 45482869 Ki > 40000 nM T77365 C8JMG7 45482870 Ki = 10400 nM T77365 C64KXS 45482874 Ki = 7030 nM T77365 CH4O5W 45483954 Ki = 6200 nM T77365 C76YLH 45483955 Ki = 2300 nM T77365 CNYS32 45483959 Ki = 3540 nM T77365 C8PFI3 45483960 Ki = 550 nM T77365 C48EWA 45483962 Ki = 277 nM T77365 CM08CA 45483963 Ki = 979 nM T77365 COT4E6 45483964 Ki = 766 nM T77365 CG50QU 45483965 Ki = 890 nM T77365 CU6XT8 45483968 Ki = 4730 nM T77365 C1LM8Y 45486932 Ki = 1340 nM T77365 C3QU2C 45487384 IC50 > 5000 nM T77365 CPCD97 46175652 IC50 > 50000 nM T77365 CD30NG 46175736 IC50 > 50000 nM T77365 C8GLI6 46175737 IC50 > 50000 nM T77365 C15UPZ 46175738 IC50 > 50000 nM T77365 CQRB27 46175914 IC50 > 50000 nM T77365 CQ9NB4 46176000 IC50 > 50000 nM T77365 CRE07N 46205479 Ki = 121 nM T77365 C5CV8H 46205480 Ki = 355 nM T77365 C5GM2E 46205481 Ki = 2020 nM T77365 C7YD4H 46205482 Ki = 1500 nM T77365 C1MS4I 46205483 Ki = 1190 nM T77365 CG60ME 46205484 Ki = 9650 nM T77365 C4B5NU 46205485 Ki = 83.8 nM T77365 CQK0G9 46205805 Ki = 843 nM T77365 CLW1U9 46205806 Ki = 127 nM T77365 CRS91E 46205807 Ki = 2180 nM T77365 CT8E0B 46205808 Ki > 30000 nM T77365 C5EZ8J 46205809 Ki = 1400 nM T77365 CS3MD6 46205810 Ki = 324 nM T77365 CLAP45 46206128 Ki > 100000 nM T77365 CK85FB 46206129 Ki > 100000 nM T77365 CTZ2J4 46206130 Ki > 100000 nM T77365 CV1HG3 46206131 Ki > 100000 nM T77365 C0XJ1G 46206132 Ki > 100000 nM T77365 CT4C0Q 46206133 Ki > 10000 nM T77365 C9TY8Z 46206464 Ki > 10000 nM T77365 COIG13 46206465 Ki = 963 nM T77365 C5NGI1 46206466 Ki > 100000 nM T77365 CYZ9G2 46206467 Ki = 778 nM T77365 C8JDB5 46206468 Ki = 2540 nM T77365 C45TYC 46206469 Ki = 8320 nM T77365 CHO5B4 46206809 Ki > 100000 nM T77365 CDS62V 46206810 Ki > 100000 nM T77365 C7RP3G 46206811 Ki = 23900 nM T77365 CMIE96 46213946 IC50 = 28 nM T77365 C5Q3GH 46225677 Ki = 586 nM T77365 C9X6TQ 46225735 Ki = 6.5 nM T77365 COZQ07 46226791 Ki = 161 nM T77365 C3GC7Q 46226793 Ki = 108 nM T77365 C5TUH7 46226812 Ki = 57.6 nM T77365 C25QHA 46226822 Ki = 15.2 nM T77365 CSR2C5 46226840 Ki = 1600 nM T77365 C01JNB 46226841 Ki = 122 nM T77365 C9E3JO 46227950 Ki = 457.09 nM T77365 CGC6Z1 46227951 Ki = 489.78 nM T77365 C3R1YJ 46227952 Ki = 380.19 nM T77365 C82AHQ 46227957 Ki = 2089.3 nM T77365 CFPO49 46227958 Ki = 1230.27 nM T77365 CHT97D 46227959 Ki = 912.01 nM T77365 C95RAL 46227973 Ki = 691.83 nM T77365 CFKX20 46227974 Ki = 489.78 nM T77365 CK1A0T 46227980 Ki = 1445.44 nM T77365 CHO9J8 46227984 Ki = 147.91 nM T77365 CB83SH 46227993 Ki = 426.58 nM T77365 CP5K0S 46227994 Ki = 1047.13 nM T77365 CFGA04 46227995 Ki = 891.25 nM T77365 CUD8P1 46228002 Ki = 524.81 nM T77365 C2MW6U 46228003 Ki = 363.08 nM T77365 C8VE7J 46228004 Ki = 1819.7 nM T77365 C4PSD1 46228006 Ki = 89.13 nM T77365 C30RBH 46228011 Ki = 416.87 nM T77365 CBV1C2 46228018 Ki = 104.71 nM T77365 CXM4R0 46228022 Ki = 309.03 nM T77365 CE42MY 46228023 Ki = 309.03 nM T77365 CB5OQ0 46228057 Ki = 446.68 nM T77365 CT61WP 46228058 Ki = 239.88 nM T77365 C5C0LN 46228971 Ki = 6250 nM T77365 CAD9G4 46229141 Ki = 100.4 nM T77365 CJ8CU7 46229272 IC50 > 100 nM T77365 CYP95V 46230103 Ki = 27 nM T77365 C84FJI 46230104 Ki = 39 nM T77365 C4XIH8 46230150 Ki = 702 nM T77365 C1KVY2 46230151 IC50 = 56 nM T77365 CL2U7N 46230192 Ki > 10000 nM T77365 CQ68OL 46230193 Ki = 5406 nM T77365 CA3RL7 46230194 Ki = 5491 nM T77365 C0YIT3 46230236 IC50 = 5 nM T77365 CV45DT 46230237 Ki = 4.6 nM T77365 C7EWV0 46230238 Ki = 5.2 nM T77365 CT4AE8 46230239 Ki = 16 nM T77365 C21NRT 46230240 Ki = 7.9 nM T77365 CN1ZO5 46230241 Ki = 1666 nM T77365 CYJ4I0 46230242 Ki = 5472 nM T77365 C6SQM4 46230243 Ki = 97 nM T77365 CYRI27 46230244 Ki = 146 nM T77365 CA2D1R 46230245 Ki = 38 nM T77365 C1B9ZU 46230246 Ki = 34 nM T77365 C80CWB 46230290 IC50 = 5.3 nM T77365 CL7F1S 46230291 Ki = 48 nM T77365 CHG01W 46230545 Ki = 4330 nM T77365 C4W9GM 46230546 Ki = 7040 nM T77365 CXP30Y 46230548 Ki = 6730 nM T77365 CVJ3F6 46230549 Ki = 5490 nM T77365 CJO4C3 46230552 Ki = 5740 nM T77365 COE2I7 46230553 Ki = 2440 nM T77365 CBRN59 46230554 Ki = 1630 nM T77365 C0EF4K 46230555 Ki = 7240 nM T77365 C0PG7O 46230556 Ki = 3280 nM T77365 CGZA62 46232472 Ki = 2800 nM T77365 CUH7B6 46232619 Ki = 6100 nM T77365 C7Q1YG 46232972 Ki > 100000 nM T77365 CM1H7R 46233161 Ki = 1445.44 nM T77365 CT5CF9 46233315 Ki = 3981.07 nM T77365 C8GM6X 46233347 Ki = 758.58 nM T77365 CLK4P1 46233348 Ki = 1737.8 nM T77365 C17TOR 46233377 Ki = 123.03 nM T77365 C3MCA6 46233378 Ki = 218.78 nM T77365 C8PJ7D 46233379 Ki = 177.83 nM T77365 CEXP72 46237805 Ki > 10000 nM T77365 C5TRP3 46237926 Ki = 121.1 nM T77365 C9GM2W 46237927 Ki = 1000 nM T77365 CG57HC 46237928 Ki = 728.1 nM T77365 C0Z1AL 46237929 Ki = 3179 nM T77365 CCJ09W 46237930 Ki = 886 nM T77365 CN36TB 46237931 Ki > 10000 nM T77365 C7US4A 46237932 Ki > 10000 nM T77365 CX5RZ3 46238063 Ki > 10000 nM T77365 CB6P5J 46238064 Ki = 180.6 nM T77365 C5LKY8 46238065 Ki > 10000 nM T77365 CM6K9V 46238066 Ki > 10000 nM T77365 CMD67R 46238067 Ki > 10000 nM T77365 C9S4VL 46238068 Ki > 10000 nM T77365 C7DPI4 46238208 Ki > 10000 nM T77365 CP9QS1 46238209 Ki = 227 nM T77365 CI3S2V 46238210 Ki = 1136 nM T77365 CS4T7D 46238211 Ki = 314 nM T77365 CD60TM 46238212 Ki = 96 nM T77365 CX6OK2 46238213 Ki > 10000 nM T77365 CAY7J1 46238338 Ki > 10000 nM T77365 C6PQR8 46238339 Ki > 10000 nM T77365 CWS95Q 46238340 Ki > 10000 nM T77365 CW41JP 46238341 Ki = 4900 nM T77365 CO5J9W 46238636 IC50 = 33 nM T77365 CES60L 46238684 IC50 = 33 nM T77365 C5H9JS 46238686 IC50 = 22 nM T77365 CXI4A9 46238694 IC50 = 333 nM T77365 C0I1XV 46238729 IC50 = 168 nM T77365 C3L9OR 46240228 IC50 = 41 nM T77365 C9O2KM 46391804 Ki > 100000 nM T77365 CKGM09 46837704 Ki = 6456.54 nM T77365 CW49MF 46846866 Ki = 3 nM T77365 C4QBV9 46846868 Ki = 12 nM T77365 C71GBF 46861670 Ki > 10000 nM T77365 CLH9D6 46861672 Ki > 10000 nM T77365 C9GCO1 46861768 Ki = 3.3 nM T77365 C9X2WT 46861769 Ki = 2.5 nM T77365 C0RFZ6 46861770 Ki = 3.6 nM T77365 CDCK67 46861780 Ki = 4.4 nM T77365 CK8D9S 46861781 Ki = 2.7 nM T77365 CIB5U2 46861782 Ki = 11.4 nM T77365 CC50RJ 46863665 Ki = 4.1 nM T77365 CU09WX 46865328 Ki = 0.38 nM T77365 CB62WH 46865329 Ki = 0.12 nM T77365 CHY8V9 46865434 Ki = 0.016 nM T77365 C5QXL9 46866591 Ki = 30 nM T77365 C8VJ9K 46866592 Ki = 239 nM T77365 CK9AU5 46866593 Ki = 150 nM T77365 CM4B3L 46874149 Ki = 1330 nM T77365 COPM34 46874262 Ki = 1533 nM T77365 CA2S6O 46875997 Ki = 4450 nM T77365 CC5OH2 46876751 Ki > 1000 nM T77365 CC7B4U 46877219 Ki > 1000 nM T77365 CY6S3U 46877262 Ki > 1000 nM T77365 CT82OL 46877263 Ki > 1000 nM T77365 CKUF93 46877269 Ki > 1000 nM T77365 CLU0A9 46877270 Ki > 1000 nM T77365 C5D2NU 46877277 Ki > 1000 nM T77365 CCH83Y 46877278 Ki > 1000 nM T77365 CP3RO7 46877284 Ki > 1000 nM T77365 CHI72K 46877285 Ki > 1000 nM T77365 C3FJZ9 46877286 Ki > 1000 nM T77365 CWD63T 46877289 Ki > 1000 nM T77365 COJW51 46877298 Ki > 1000 nM T77365 C5MB9D 46877311 Ki > 1000 nM T77365 CJ6LH9 46877313 Ki > 1000 nM T77365 CFV06U 46877320 Ki > 1000 nM T77365 C8H2FW 46877321 Ki > 1000 nM T77365 C8C6VB 46877325 Ki > 1000 nM T77365 C3F5EW 46877333 Ki > 1000 nM T77365 CNYJ02 46877335 Ki > 1000 nM T77365 C50XUB 46880372 Ki = 35 nM T77365 CZJ2V5 46880373 Ki = 12 nM T77365 CL8UH3 46880375 Ki = 147 nM T77365 CQ93IM 46880419 Ki = 11 nM T77365 CMCX40 46880420 Ki = 302 nM T77365 C7P6TS 46880421 Ki = 813 nM T77365 CKB31F 46880422 Ki = 1359 nM T77365 CH5B6C 46880424 Ki = 181 nM T77365 CB9TI2 46880470 Ki = 635 nM T77365 C46AYO 46880471 Ki = 1373 nM T77365 CSXZ76 46880473 Ki = 1440 nM T77365 COQ7X3 46880474 Ki = 61 nM T77365 C2SM9Q 46880475 Ki = 57 nM T77365 CV10FQ 46880506 Ki = 286 nM T77365 CMP72U 46880507 Ki = 39 nM T77365 CM36IE 46880508 Ki = 862 nM T77365 CS2X0C 46880509 Ki = 1465 nM T77365 C61JDB 46880510 Ki = 163 nM T77365 C1TG8M 46882994 IC50 = 6685 nM T77365 CO0P9H 46882995 IC50 = 7847 nM T77365 C95IFA 46882996 IC50 = 3852 nM T77365 C2F0IA 46882997 IC50 = 220 nM T77365 C14OFC 46882998 IC50 = 126 nM T77365 C97CLT 46883039 IC50 > 10000 nM T77365 CD50FZ 46883040 IC50 = 7146 nM T77365 CQT47C 46883041 IC50 = 1077 nM T77365 CYUD90 46883042 IC50 = 186 nM T77365 CA4O8S 46883043 IC50 = 990 nM T77365 CE12TM 46883070 IC50 = 116 nM T77365 C19PUS 46883071 IC50 = 161 nM T77365 C93JQZ 46883072 IC50 = 351 nM T77365 C5UOJ7 46883073 IC50 = 177 nM T77365 CJG6K1 46883074 IC50 = 2271 nM T77365 CKQG17 46883106 IC50 = 118 nM T77365 C12NEL 46883107 IC50 = 99 nM T77365 CBZ74M 46883108 IC50 = 1541 nM T77365 CXQW19 46883109 IC50 = 1252 nM T77365 C3T4YP 46883110 IC50 = 51 nM T77365 C4M6IK 46883155 IC50 = 405 nM T77365 CJ1L0R 46883156 IC50 = 732 nM T77365 CD6EW1 46883157 IC50 = 1715 nM T77365 CXA5L7 46883158 IC50 = 1619 nM T77365 CSK8A5 46883159 IC50 = 442 nM T77365 CS31KC 46883205 IC50 = 637 nM T77365 CM0Z4K 46883206 IC50 = 1168 nM T77365 CG4J3B 46883207 IC50 = 1942 nM T77365 CJ57AD 46883208 IC50 = 62 nM T77365 CGZ31A 46885889 Ki = 3.56 nM T77365 CB0W8K 46885950 Ki = 1.1 nM T77365 CP9G2T 46885951 Ki = 2.02 nM T77365 CU7A4P 46885952 Ki = 0.152 nM T77365 C7Y8UP 46885953 Ki = 0.038 nM T77365 C8D1QP 46885990 Ki = 0.7 nM T77365 C0TGQ9 46885991 Ki = 0.57 nM T77365 C4ELG9 46885992 Ki = 0.0082 nM T77365 C1K9IJ 46886592 IC50 = 45 nM T77365 C7JC1V 46886593 IC50 = 10 nM T77365 CUTZ94 46886594 IC50 = 305 nM T77365 C3Z0AW 46886595 IC50 = 10 nM T77365 CR69BT 46886596 IC50 = 6 nM T77365 CNK98E 46886597 IC50 = 4 nM T77365 CZPO78 46886598 IC50 = 5 nM T77365 C01EXI 46887114 Ki = 600 nM T77365 CZY7M9 46887155 Ki = 400 nM T77365 C5EGF2 46887668 Ki > 10000 nM T77365 C0S7BL 46887669 Ki > 10000 nM T77365 CA41WQ 46887671 Ki > 10000 nM T77365 C0TF5V 46887672 Ki > 10000 nM T77365 CQP3K6 46887673 Ki > 10000 nM T77365 C9PS5C 46888223 Ki > 10000 nM T77365 C6NCF2 46888282 Ki > 10000 nM T77365 C2SX3E 46888356 Ki > 10000 nM T77365 C7YGA4 46888359 Ki > 10000 nM T77365 CZXY41 46888782 Ki = 35.3 nM T77365 C0ZI2J 46888783 Ki = 18.1 nM T77365 C3PO0V 46888784 Ki = 19.3 nM T77365 CNJ6O8 46888821 Ki = 35.1 nM T77365 CM4KX9 46888822 Ki = 4.7 nM T77365 CS6YQ2 46888823 Ki = 0.9 nM T77365 C7F0ZH 46888824 Ki = 0.9 nM T77365 CPU7O1 46888850 Ki = 3.1 nM T77365 CR76TD 46888851 Ki = 12.5 nM T77365 CP3M2V 46888852 Ki = 4.9 nM T77365 CZY0H4 46888879 Ki = 2.9 nM T77365 CXEM23 46888880 Ki = 23.2 nM T77365 C6PEB7 46888881 Ki = 10 nM T77365 C1DOU2 46888889 Ki = 0.2 nM T77365 CY9HA1 46888890 Ki = 10.5 nM T77365 C27AJV 46888923 Ki = 76.6 nM T77365 CLA81S 46888924 Ki = 117 nM T77365 CQK1W2 46888929 Ki = 0.5 nM T77365 CJI92H 46888930 Ki = 4.6 nM T77365 CW3GP5 46888987 Ki = 32.5 nM T77365 CJ40AW 46888988 Ki = 40.1 nM T77365 C3HTX6 46888989 Ki = 18.3 nM T77365 CI6WP9 46888990 Ki = 14.3 nM T77365 CGE3Q5 46888991 Ki = 11.3 nM T77365 CLVB51 46889017 Ki = 7.9 nM T77365 C6LOJ5 46889018 Ki = 8.6 nM T77365 CZD9E7 46889019 Ki = 3.8 nM T77365 CW8UG0 46889042 Ki = 5.4 nM T77365 CMK23N 46889043 Ki = 11.3 nM T77365 CFJG37 46889044 Ki = 5.3 nM T77365 C5B2MH 46889068 Ki = 5.4 nM T77365 CP87LM 46889069 Ki = 3 nM T77365 CSFA02 46889070 Ki = 9.9 nM T77365 CG1YE0 46889071 Ki = 9.3 nM T77365 CP0JK9 46889095 Ki = 29.8 nM T77365 C45LRI 46889096 Ki = 12.9 nM T77365 C4P8EK 46889097 Ki = 5.9 nM T77365 CN51XZ 46889098 Ki = 1 nM T77365 CA3G2B 46889125 Ki = 4.1 nM T77365 CUZW61 46889126 Ki = 12.8 nM T77365 CIU27M 46889127 Ki = 7.8 nM T77365 CT6F8I 46889171 Ki = 12.4 nM T77365 C1SKA9 46889172 Ki = 7.8 nM T77365 C4HFX9 46889173 Ki = 13.5 nM T77365 CFP4E5 46889174 Ki = 28.4 nM T77365 CS4L1B 46889205 Ki = 18.6 nM T77365 C0ZJ5W 46889206 Ki = 16.8 nM T77365 CQSP94 46889207 Ki = 32.5 nM T77365 CE43BM 46889228 Ki = 11.1 nM T77365 C7PO4J 46889229 Ki = 14.9 nM T77365 CF7I9L 46889230 Ki = 32.1 nM T77365 CI67DB 46889231 Ki = 20.7 nM T77365 CG1AU4 46889252 Ki = 17.3 nM T77365 C83ZFB 46889253 Ki = 37.3 nM T77365 CMJ61R 46889254 Ki = 7.9 nM T77365 C9NHC7 46889255 Ki = 50.6 nM T77365 C4O0IB 46889256 Ki = 13.7 nM T77365 CUFE02 46893147 EC50 = 460 nM T77365 C3JCB1 46911060 Ki = 51 nM T77365 C1LCB2 46912311 Ki = 53 nM T77365 C3H4CM 46912312 Ki = 19 nM T77365 CNU1T6 46912313 Ki = 22 nM T77365 CDTQ70 46912314 Ki = 12 nM T77365 C1BJF7 46912315 Ki = 7.5 nM T77365 CY35KS 46943091 Ki = 2398.83 nM T77365 CJHW13 46945058 Ki = 12.4 nM T77365 C02HEX 49797747 Ki = 76 nM T77365 CC61BT 49797748 Ki = 100 nM T77365 C8HA0Y 49797749 Ki = 66 nM T77365 C6XFQ7 49797750 Ki = 80 nM T77365 CP1I3U 49797771 Ki = 77 nM T77365 CN4UQ9 49797772 Ki = 27 nM T77365 CF32QB 49797773 Ki = 71 nM T77365 CB0X1S 49797774 Ki = 46 nM T77365 C21IWV 49797793 Ki = 170 nM T77365 C4Y0JV 49797794 Ki = 50 nM T77365 C6X5LC 49797795 Ki = 92 nM T77365 CD26ZY 49797796 Ki = 15 nM T77365 CN58DG 49797797 Ki = 480 nM T77365 CY1XE9 49797825 Ki = 330 nM T77365 CXJV63 49797826 Ki = 160 nM T77365 C4JX9B 49797827 Ki = 2200 nM T77365 CXH10P 49797828 Ki = 5 nM T77365 CF0H2A 49797852 Ki = 29 nM T77365 C7SH3X 49797853 Ki = 98 nM T77365 C7DM9C 49797854 Ki = 61 nM T77365 CB87EF 49797855 Ki = 35 nM T77365 C8FD9E 49797878 Ki = 3 nM T77365 CNRX41 49797879 Ki = 18 nM T77365 CU1H3X 49797904 Ki = 41 nM T77365 CO69IE 49797905 Ki = 3 nM T77365 C9AVX7 49797906 Ki = 3 nM T77365 CSB23K 49798137 Ki = 68 nM T77365 CJ15VM 49798138 Ki = 84 nM T77365 CEC37Y 49798139 Ki = 89 nM T77365 C7P6DN 49798140 Ki = 26 nM T77365 CZIB48 49798161 Ki = 707.95 nM T77365 CJ8CH9 49863226 Ki = 400 nM T77365 C6UJI0 49864319 Ki = 220 nM T77365 CW1I8V 49864320 Ki = 460 nM T77365 C3J7QB 49864672 Ki = 62 nM T77365 C84BSL 49864673 Ki = 190 nM T77365 CIJV65 49864676 Ki = 290 nM T77365 C2GP3F 49864677 Ki = 700 nM T77365 C4OB0D 49864730 Ki = 410 nM T77365 CR14MY 49864731 Ki = 340 nM T77365 C7I2SE 49864732 Ki = 330 nM T77365 CY8B6L 49864733 Ki = 710 nM T77365 C5YQM7 49870825 Ki = 805.1 nM T77365 CFX9W2 49870826 Ki = 2115 nM T77365 CYKD61 49870828 Ki = 7365 nM T77365 C8WP4Y 49870952 Ki = 7.19 nM T77365 CE9Q3P 49870953 EC50 = 20.6 nM T77365 C8XWJ3 50899648 Ki = 12 nM T77365 C4WXE2 50925499 Ki > 10000 nM T77365 C0OQI7 50940921 Ki = 183 nM T77365 C1UMB4 50940926 Ki = 424 nM T77365 CCD60O 50940932 Ki = 1893 nM T77365 CAN28T 50940939 Ki = 647 nM T77365 CY3QD4 50940944 Ki = 201 nM T77365 CUS54E 50940957 Ki = 1334 nM T77365 C9LV4F 50940960 Ki = 73.8 nM T77365 CIZ5W0 50940962 Ki = 3345 nM T77365 CD1U2T 50940964 Ki = 8.1 nM T77365 CY7J8X 50940965 Ki = 24.6 nM T77365 CLY1D0 50940966 Ki = 74 nM T77365 C13NAI 50940967 Ki = 39.8 nM T77365 CZ4WU9 50940972 Ki = 429 nM T77365 C7CH3U 50940974 Ki = 103 nM T77365 CJC06P 50940976 Ki = 2541 nM T77365 CB5TZ6 50940978 Ki = 6.4 nM T77365 CMF2S3 50940979 Ki = 114 nM T77365 C5H8FK 50940980 Ki = 82.8 nM T77365 CW76LB 50940981 Ki = 63.5 nM T77365 CEZM81 50940986 Ki = 1829 nM T77365 CPB75Y 50940989 Ki = 142 nM T77365 C1B7TN 50941005 Ki = 5.7 nM T77365 CLE1G9 50941006 Ki = 153 nM T77365 CY4W7P 50941007 Ki = 544 nM T77365 C2J0GZ 51039221 Ki = 27.3 nM T77365 CS36WH 51039222 Ki = 11.1 nM T77365 CPY2L4 51039223 Ki = 11.5 nM T77365 CUB5G9 51040798 Ki = 933 nM T77365 CZ2NF4 51050120 Ki = 28 nM T77365 CM6T0R 51050123 Ki = 110 nM T77365 C30EZP 51050124 Ki = 180 nM T77365 COM32L 51050226 Ki = 32 nM T77365 C3ACR2 51050227 Ki = 12 nM T77365 C8P3IT 51050841 Ki = 21 nM T77365 COFS19 51050842 Ki = 153 nM T77365 C96NLK 51050843 Ki = 40.9 nM T77365 C32PZT 51050844 Ki = 69.7 nM T77365 CYBC20 51050845 Ki = 38.6 nM T77365 CO3N1B 51050939 Ki = 44.7 nM T77365 CGCI34 51050940 Ki = 17.8 nM T77365 C35FWV 51050941 Ki = 52.3 nM T77365 CBX3Q5 51050942 Ki = 86.2 nM T77365 C35OZM 51050943 Ki = 124 nM T77365 CRPE85 51050944 Ki = 94.8 nM T77365 CE2ZF4 51051035 Ki = 66.2 nM T77365 C67BTI 51051036 Ki = 282 nM T77365 C2WTK7 51051037 Ki = 212 nM T77365 CT5Z6U 51051038 Ki = 348 nM T77365 C9U0PR 51051039 Ki = 7680 nM T77365 CG5P0M 51051040 Ki = 39.1 nM T77365 C2F7LS 51051138 Ki = 567 nM T77365 C37NQZ 51051140 Ki = 16.9 nM T77365 C72UZF 51051141 Ki = 270 nM T77365 CP4Q8Y 51051143 Ki = 90.1 nM T77365 CK12HU 51051145 Ki = 92.9 nM T77365 C6BN9V 51051146 Ki = 58.4 nM T77365 CTZ4H6 51051245 Ki = 4360 nM T77365 CHX3O5 51051246 Ki = 38200 nM T77365 CVBO13 51051248 Ki = 1000 nM T77365 CR2TW4 51051249 Ki = 160 nM T77365 C1DB8M 51051251 Ki = 44.1 nM T77365 C8Z0NV 52912216 Ki > 10000 nM T77365 C8SX6V 52933926 Ki = 2000 nM T77365 CS8FG1 52940825 Ki = 35 nM T77365 CU2SW9 52940875 Ki = 25 nM T77365 CCE8X6 52940891 Ki = 37 nM T77365 CI82OJ 52940945 Ki = 16 nM T77365 C8VZ2U 52940999 Ki > 10000 nM T77365 CT53UX 52941201 Ki > 10000 nM T77365 CSGQ69 52941244 Ki > 10000 nM T77365 CCL3P4 52941437 Ki = 308 nM T77365 C9H3FM 52941478 IC50 > 50000 nM T77365 C9O5BW 52941481 Ki = 23.9 nM T77365 C71HWB 52941597 Ki > 10000 nM T77365 CF72VX 52942026 Ki = 92 nM T77365 CE4L6P 52942060 Ki = 123 nM T77365 C2VJ8B 52942091 Ki = 51 nM T77365 CA60PY 52942205 Ki = 2.5 nM T77365 C8XKR4 52942290 Ki = 6770 nM T77365 CQF4X5 52942334 Ki = 5190 nM T77365 C3J6FO 52942359 Ki > 10000 nM T77365 CCJP23 52942475 Ki = 1080 nM T77365 CV8EW1 52942501 Ki = 878 nM T77365 CO31WJ 52942623 Ki = 9 nM T77365 CX5S2B 52942735 Ki = 45.7 nM T77365 CI0A6Z 52942905 Ki = 3300 nM T77365 CQ1M9B 52943279 Ki = 904 nM T77365 CL4IQ3 52943294 Ki = 233 nM T77365 C2T1RZ 52943351 Ki = 13 nM T77365 CV6JI9 52943490 Ki > 10000 nM T77365 C2BJZ3 52943652 Ki = 2439 nM T77365 C4WJ3T 52943806 Ki = 22.1 nM T77365 CTMG40 52944560 Ki = 1670 nM T77365 CT0Y9I 52944659 Ki = 3150 nM T77365 CEO93J 52944665 Ki = 67.9 nM T77365 C5I4BV 52944930 Ki = 3509 nM T77365 CVB60F 52945006 Ki > 10000 nM T77365 C2H9AY 52945064 Ki > 10000 nM T77365 CJAY05 52945098 Ki > 10000 nM T77365 CY8LW4 52945120 Ki = 78.9 nM T77365 C45SQC 52945195 Ki = 1925 nM T77365 CV1Z6M 52945246 Ki = 179 nM T77365 CUL5Y9 52945717 Ki = 11 nM T77365 CHT4Z6 52946113 Ki > 10000 nM T77365 CX9G3T 52946114 Ki > 10000 nM T77365 CK76UG 52946159 Ki > 10000 nM T77365 CEFW97 52946211 IC50 > 50000 nM T77365 CF5K9X 52946213 Ki = 13.3 nM T77365 CUA1O9 52946453 Ki > 10000 nM T77365 C0APZ7 52946949 Ki = 1220 nM T77365 C28VAP 52947301 Ki > 10000 nM T77365 CH54XQ 52947440 Ki = 11.7 nM T77365 C7HY0V 52947452 Ki > 10000 nM T77365 CV9D1Y 52947525 IC50 = 5500 nM T77365 CE6C4T 52947707 Ki = 2590 nM T77365 C8UGP7 52947752 Ki = 9.6 nM T77365 C2FZK0 52947764 Ki = 14.4 nM T77365 C38OQX 52948144 Ki = 147 nM T77365 CV08MP 52948170 Ki = 1100 nM T77365 C8Q3UH 52948332 Ki = 1760 nM T77365 C6JN5H 52948418 Ki = 2490 nM T77365 C4KA6Y 52948671 Ki > 10000 nM T77365 COW0J3 52948763 Ki > 10000 nM T77365 C3B9OG 52948788 IC50 > 50000 nM T77365 C7TI2R 52948915 Ki > 10000 nM T77365 C28MQF 52948949 Ki > 10000 nM T77365 CQ91YN 52948995 IC50 > 50000 nM T77365 C5D2JP 52949382 Ki = 7.7 nM T77365 CHAX52 52949423 Ki = 325 nM T77365 CLHR35 52949461 Ki = 2430 nM T77365 CK6R3J 52949519 Ki = 43.9 nM T77365 C6ZXI9 52949641 Ki = 572.1 nM T77365 C2MAQ9 52949644 Ki = 772.5 nM T77365 C67NOY 52949655 Ki = 501.2 nM T77365 CE8F3G 52949755 Ki > 10000 nM T77365 CE3XQ7 52949772 Ki > 10000 nM T77365 CL6K9M 52949999 Ki > 10000 nM T77365 C74BRO 52950000 Ki > 10000 nM T77365 CHM1G6 52950027 Ki > 10000 nM T77365 CQAP62 52950040 Ki = 1460 nM T77365 C3JEO8 52950206 Ki > 10000 nM T77365 C7DWU2 53131655 Ki = 36307.81 nM T77365 CRB59S 53242165 Ki = 530 nM T77365 CI35WL 53248698 Ki = 2040 nM T77365 CDS80Q 53248700 Ki = 210 nM T77365 CJZ98W 53318744 Ki = 145 nM T77365 CA91KC 53322692 Ki = 408 nM T77365 CH7O8A 53324032 Ki = 101 nM T77365 CY04CM 53325341 Ki = 634 nM T77365 CN51SY 53348048 Ki > 10000 nM T77365 C7NOK1 53353232 Ki = 21.38 nM T77365 CIVP28 53354521 Ki = 51.29 nM T77365 CIAO19 53354627 Ki = 16 nM T77365 CH6X9F 53354632 Ki = 3.981 nM T77365 C45VUI 53354728 Ki = 41 nM T77365 CL3P8I 53394567 Ki = 7730 nM T77365 CUO97T 54577823 Ki = 417 nM T77365 CZQ2H9 54580150 Ki = 1000 nM T77365 C9LU8J 54580623 Ki > 100000 nM T77365 CT1CO5 54580654 Ki = 75.4 nM T77365 CY4W3B 54580983 Ki > 1300 nM T77365 CIWP03 54581016 Ki > 1500 nM T77365 C84FJX 54581142 Ki = 110 nM T77365 CSX07T 54581143 Ki = 31 nM T77365 CX3Y6L 54581663 Ki = 53.6 nM T77365 C9PI3B 54582022 Ki = 1 nM T77365 C85ZXD 54582166 Ki = 81 nM T77365 C2C8MB 54582167 Ki = 280 nM T77365 C5RQJ9 54582654 Ki = 10.7 nM T77365 CHDV60 54583133 Ki = 180 nM T77365 CHXE36 54583615 Ki = 96 nM T77365 C08HKQ 54583616 Ki = 330 nM T77365 CSF9W8 54583714 Ki = 220 nM T77365 CS8LX5 54583961 Ki > 1500 nM T77365 CM4D3E 54583968 Ki > 1300 nM T77365 CY52BQ 54583969 Ki > 1300 nM T77365 CS6O9E 54584124 Ki = 230 nM T77365 C7CWY9 54584125 Ki = 1040 nM T77365 CP04UN 54584599 Ki = 6.8 nM T77365 C3N7RC 54585057 Ki = 52 nM T77365 CO7IC0 54585058 Ki = 240 nM T77365 CKCD81 54585511 Ki = 55000 nM T77365 CVG5I1 54585877 Ki = 8.7 nM T77365 C02CVB 54586036 Ki = 710 nM T77365 C4SZ1B 54586516 Ki = 357 nM T77365 CT80FJ 54586843 Ki = 556 nM T77365 CNA0S3 54586844 Ki = 15.6 nM T77365 C6IV3L 54587015 Ki = 600 nM T77365 CR3QM0 54587363 Ki = 1700 nM T77365 CP89KE 54587624 Ki = 15.1 nM T77365 CSL08D 54587662 Ki = 3090 nM T77365 C83VFS 54754508 Ki = 1460 nM T77365 C40IVD 54768079 Ki = 1160 nM T77365 C1UW4E 54768080 Ki > 10000 nM T77365 C4JA9T 54768112 Ki > 10000 nM T77365 C2JPC3 54768115 Ki = 2400 nM T77365 CL5SE3 54768601 Ki = 3270 nM T77365 C6SYD1 54768602 Ki = 306 nM T77365 CX9A4R 54768635 Ki = 847 nM T77365 C3HNS6 54768636 Ki = 21900 nM T77365 C91PGO 56603115 Ki > 10000 nM T77365 CB7T1O 56627882 EC50 = 3.84 nM T77365 C6WSF9 56657920 Ki = 6930 nM T77365 CD7C2P 56661442 Ki = 19400 nM T77365 C2FI4U 56661443 Ki = 25200 nM T77365 CZ6I4O 56662964 Ki = 750 nM T77365 CVLM74 56664888 Ki > 100000 nM T77365 CBQS24 56668308 Ki = 4040 nM T77365 CYNJ53 56668410 Ki > 30000 nM T77365 CWM34N 56668411 Ki = 36000 nM T77365 CSJ34D 56668412 Ki > 30000 nM T77365 C98FPH 56671922 Ki > 100000 nM T77365 CD6C0P 56675199 Ki > 100000 nM T77365 CH8YR5 56675200 Ki = 614 nM T77365 CUJ34X 56675201 Ki = 571 nM T77365 CK3AZ9 56675297 Ki = 987 nM T77365 C58FTQ 56675298 Ki = 2360 nM T77365 C7TNW9 56675299 Ki = 5930 nM T77365 CDN69Q 56678498 Ki > 10000 nM T77365 C13UZX 56678638 Ki = 1060 nM T77365 CM04LK 56678639 Ki > 30000 nM T77365 CVP0A9 56681843 Ki = 8400 nM T77365 C02DIY 56838950 EC50 = 117 nM T77365 CYS17U 56844240 Ki = 7.762 nM T77365 COY13J 56924646 Ki > 1000 nM T77365 C86NML 56935713 Ki = 4700 nM T77365 CF60KW 56943766 Ki = 0.42 nM T77365 C5CG7W 56943866 Ki = 0.07 nM T77365 CB0ML9 56943867 Ki = 0.21 nM T77365 CTSP76 56943869 Ki = 0.4 nM T77365 CIX25P 56943870 Ki = 1.1 nM T77365 C47RTV 56943872 Ki = 1.2 nM T77365 CTWN13 56943964 Ki = 0.06 nM T77365 CXI7C1 56943965 Ki = 0.5 nM T77365 CK0WV9 56943966 Ki = 4.5 nM T77365 C4AL1U 56943967 Ki = 0.7 nM T77365 C2O4GP 56944062 Ki = 0.25 nM T77365 CK42GD 56944063 Ki = 0.9 nM T77365 CZJ31A 56944261 Ki = 0.5 nM T77365 C8TZ4I 56944263 Ki = 0.3 nM T77365 CKN1X7 56944264 Ki = 0.4 nM T77365 CY87XN 56944265 Ki = 3.1 nM T77365 CS9HN3 56944354 Ki = 0.9 nM T77365 CUCF59 56944358 Ki = 0.2 nM T77365 CJAN-69 56944443 Ki = 0.26 nM T77365 CW4T7L 56944733 Ki = 0.27 nM T77365 C1L2ZK 56944736 Ki = 0.15 nM T77365 CB7I4R 56945639 Ki = 63.2 nM T77365 C9XFM7 56945648 Ki = 160 nM T77365 CCK34B 56945649 Ki = 84.3 nM T77365 C3WC9H 56945650 Ki = 87.2 nM T77365 C0C8EV 56945751 Ki = 2160 nM T77365 CD54JK 56945753 Ki = 3730 nM T77365 CMP74W 56945754 Ki = 3910 nM T77365 C5DT0Z 56945768 Ki = 130 nM T77365 CU4C5D 56945769 Ki = 180 nM T77365 CR1YL9 56945770 Ki = 110 nM T77365 CPA2Z6 56945771 Ki = 100 nM T77365 C9HK5A 56945866 Ki = 4890 nM T77365 CMAO83 56945867 Ki = 178 nM T77365 CKZE52 56945888 Ki = 50 nM T77365 C9VLJ0 56945889 Ki = 63.7 nM T77365 CRF5J8 56945890 Ki = 34 nM T77365 CX3W2C 56945891 Ki = 71.7 nM T77365 CD4ZW9 56945994 Ki = 130 nM T77365 CI0Q2T 56945995 Ki = 110 nM T77365 CR5AJ1 56945996 Ki = 40 nM T77365 CH1JR4 56950235 Ki = 500 nM T77365 CXB8Z6 56951623 Ki = 960 nM T77365 C9F7YE 56954252 Ki = 0.1 nM T77365 CTXB04 56954253 Ki = 0.5 nM T77365 C70KFB 56954254 Ki = 1.6 nM T77365 CL56UR 56954333 Ki = 3.1 nM T77365 CLTD39 56954334 Ki = 1.4 nM T77365 CIJN02 56954335 Ki = 1.3 nM T77365 CH5A4T 56954336 Ki = 0.7 nM T77365 CH3GM5 56964225 Ki = 3.467 nM T77365 C9T1XQ 56964459 Ki > 10000 nM T77365 CY1IG3 56964460 Ki = 50.6 nM T77365 CZ42XV 56964461 Ki > 10000 nM T77365 CC50SG 56964576 Ki > 10000 nM T77365 CHR8L5 57325914 Ki = 15.8 nM T77365 C7SRT3 57325915 Ki > 10000 nM T77365 CPJG73 57327005 Ki = 0.56 nM T77365 CREU79 57328471 Ki > 100000 nM T77365 C8JY3E 57384287 EC50 = 45 nM T77365 CYSA75 57384288 EC50 = 14 nM T77365 CDN54M 57384289 EC50 = 6.6 nM T77365 CA63RT 57384543 EC50 = 366 nM T77365 CW63IC 57384544 EC50 = 712 nM T77365 CCPY02 57385043 EC50 = 89.7 nM T77365 CKO3L1 57387337 EC50 = 5.6 nM T77365 C8X7MO 57387594 EC50 = 0.85 nM T77365 C6XKL9 57387596 EC50 = 2.02 nM T77365 C7XW0T 57387822 EC50 = 2242 nM T77365 CT1R6Q 57387824 EC50 = 14 nM T77365 C01AHY 57387825 EC50 = 42 nM T77365 CNL3P2 57388054 EC50 = 66 nM T77365 CK7R6O 57388055 EC50 = 6.3 nM T77365 CMBN74 57388056 EC50 = 30.9 nM T77365 C1BAX6 57391653 Ki = 50 nM T77365 C45GCN 57391694 Ki = 42 nM T77365 C03HUE 57391695 Ki = 119 nM T77365 CJF61Z 57391696 Ki > 1000 nM T77365 C13NRM 57392607 Ki = 168 nM T77365 CC3X7G 57393433 Ki = 626 nM T77365 C1B3QM 57393434 Ki > 1000 nM T77365 C8ZX4L 57393435 Ki > 1000 nM T77365 CVO2P8 57395120 Ki = 200 nM T77365 C9VWH7 57395161 Ki > 1000 nM T77365 CJM7E8 57395162 Ki = 122 nM T77365 CEQR05 57395163 Ki = 68 nM T77365 CDP13M 57395164 Ki = 222 nM T77365 CDJ6W2 57396128 Ki = 2.3 nM T77365 CSTG21 57396888 Ki = 3.9 nM T77365 CWX64M 57396935 Ki = 3.6 nM T77365 CC52TB 57396936 Ki = 17 nM T77365 C1WT0H 57396937 Ki > 1000 nM T77365 CD6JT5 57398641 Ki = 30 nM T77365 CHC8U6 57398676 Ki = 11 nM T77365 C1J3DG 57400352 Ki = 12 nM T77365 CNRY34 57400353 Ki = 208 nM T77365 CIX58U 57402117 Ki = 20 nM T77365 CLCX61 57402118 Ki = 148 nM T77365 CBMP08 57402160 Ki = 130 nM T77365 C58APE 57402161 Ki = 8.1 nM T77365 CKB51R 57402162 Ki = 672 nM T77365 CQK46U 57402163 Ki > 1000 nM T77365 CYHD10 57403904 Ki = 20 nM T77365 CD2NO5 57403905 Ki = 9.2 nM T77365 C05DRY 57429649 Ki = 57 nM T77365 CX1S2Q 57523212 Ki = 1740 nM T77365 CQAW53 57523252 Ki = 3110 nM T77365 CR78ZP 57523655 Ki = 1270 nM T77365 CP9JX0 57523691 Ki = 5300 nM T77365 C8J6OD 58522807 Ki = 4 nM T77365 C1HU4O 59011969 Ki = 1500 nM T77365 CY0J5M 59276682 Ki = 19.7 nM T77365 CB31TY 59276704 Ki = 610 nM T77365 C92ZHB 59276711 Ki = 110 nM T77365 C1EWD7 59277997 Ki = 109 nM T77365 CF60BK 59277999 Ki > 168 nM T77365 C5G2RH 60154738 Ki = 1137 nM T77365 C4U7BI 60154739 Ki = 2813 nM T77365 CU3R2Q 60154740 Ki > 5000 nM T77365 CJ57XU 60154742 Ki = 1856 nM T77365 CUK15D 60154835 Ki = 1282 nM T77365 CK7VH4 60154837 Ki > 5000 nM T77365 C3PO4T 60155712 Ki > 5000 nM T77365 CJB03P 60155713 Ki > 5000 nM T77365 C6W8XE 60155714 Ki = 1193 nM T77365 CN03ZC 60155715 Ki = 1423 nM T77365 CEZ4V5 60155716 Ki = 789 nM T77365 C1ZXO7 60155796 Ki = 526 nM T77365 CZRU45 60155797 Ki > 5000 nM T77365 C8GZ3V 60155798 Ki > 5000 nM T77365 CXLO10 60155799 Ki > 5000 nM T77365 CYB1L4 60155893 Ki > 5000 nM T77365 C0B5OZ 60155894 Ki = 2223 nM T77365 CB9A6F 60155895 Ki > 5000 nM T77365 C2VPM8 60155896 Ki > 5000 nM T77365 CW7R1L 60155897 Ki > 5000 nM T77365 CP3H2Z 60156002 Ki = 1084 nM T77365 C8KU5V 60156003 Ki > 5000 nM T77365 C2LN4J 60156004 Ki > 5000 nM T77365 C8SZE0 60156005 Ki > 5000 nM T77365 CGL84Y 60156006 Ki > 5000 nM T77365 CFBG07 60156104 Ki > 5000 nM T77365 CKVJ21 60156105 Ki > 5000 nM T77365 C7L1BF 60156106 Ki = 1842 nM T77365 C38NUA 60156107 Ki = 1641 nM T77365 C87SMR 60156108 Ki = 3255 nM T77365 C2BH4J 60167948 IC50 = 30 nM T77365 C16CSN 60195998 Ki = 1600 nM T77365 CLD35T 62188326 Ki = 500 nM T77365 C1HBG4 66573213 Ki = 630.96 nM T77365 CRJ86F 66573214 Ki = 1000 nM T77365 CLM18K 66678431 Ki = 8 nM T77365 C20XJH 66892244 Ki = 486 nM T77365 CWN0X9 66892382 Ki = 36 nM T77365 CV6PW1 66892867 Ki = 192 nM T77365 C9GDP5 66894241 Ki = 124 nM T77365 C1XZV9 67364057 Ki = 15.49 nM T77365 C41MUQ 67364090 Ki = 27.54 nM T77365 CXQL59 67364157 Ki = 4.571 nM T77365 CS0D4B 67364791 Ki = 10.47 nM T77365 CW37UH 67548131 IC50 > 1000 nM T77365 C56UIN 67548175 IC50 > 1000 nM T77365 C6VKP4 67548337 IC50 = 59 nM T77365 CGXY26 67548392 IC50 = 86 nM T77365 C5U3WL 67548498 IC50 > 1000 nM T77365 C6LA7R 67548508 IC50 = 5 nM T77365 CC4Y6V 67548720 IC50 = 434 nM T77365 C8B1JS 67548983 IC50 > 1000 nM T77365 CPQ2I7 67549056 IC50 > 1000 nM T77365 C71HZU 67549086 IC50 = 105 nM T77365 C74YXW 67549097 IC50 > 1000 nM T77365 CD09WI 67549451 IC50 > 1000 nM T77365 C5M0NT 67549626 IC50 > 1000 nM T77365 C8Z7RX 67549879 IC50 > 1000 nM T77365 C17YBH 68148396 Ki > 10000 nM T77365 CQ36MR 68388533 Ki > 1000 nM T77365 C7Y2WK 68388551 Ki = 1.4 nM T77365 CDKQ62 68388674 Ki > 1000 nM T77365 C18CNK 68405754 IC50 > 1000 nM T77365 CNYS04 68405874 IC50 > 1000 nM T77365 CWEQ54 68405927 IC50 > 1000 nM T77365 C2OM6I 69029783 Ki = 53 nM T77365 CRL75S 69031481 Ki = 460 nM T77365 C0P1OR 69427076 Ki = 273 nM T77365 CXUB67 69846372 Ki = 292 nM T77365 C76KTS 69846756 Ki = 9500 nM T77365 CJ7Y1S 70676459 Ki = 3610 nM T77365 COVC42 70676460 Ki = 4910 nM T77365 C9OLG0 70676461 Ki = 1570 nM T77365 CCO40K 70676610 Ki = 3650 nM T77365 C21ANJ 70676611 Ki = 5470 nM T77365 CN38XM 70676612 Ki = 6450 nM T77365 CYTH16 70676613 Ki = 4840 nM T77365 C0VI8J 70676614 Ki = 2550 nM T77365 CZA8H7 70677100 Ki = 2230 nM T77365 CFIP08 70680953 Ki = 111 nM T77365 C46HBT 70681087 Ki = 3930 nM T77365 CIT56B 70681088 Ki = 3700 nM T77365 CE3N0Y 70681091 Ki = 7510 nM T77365 CX39FT 70681867 Ki = 398.11 nM T77365 C4ND7L 70682887 Ki = 1800 nM T77365 CS0I7Z 70682890 Ki = 94 nM T77365 C7LZO2 70683991 Ki = 316.23 nM T77365 C0XG9F 70685288 Ki = 2720 nM T77365 C7AXZ8 70686118 Ki = 1584.89 nM T77365 CN86WI 70686119 Ki = 501.19 nM T77365 CM03SU 70687435 Ki = 3020 nM T77365 CL63IQ 70687436 Ki = 4410 nM T77365 CB3D6N 70688247 Ki = 398.11 nM T77365 CAWY65 70688249 Ki = 630.96 nM T77365 C1KJD5 70689262 Ki = 1 nM T77365 C7X1UJ 70689496 Ki = 3140 nM T77365 CA4E1B 70690267 Ki = 501.19 nM T77365 CZ9S6P 70691273 Ki = 680 nM T77365 C58QIA 70691614 Ki = 4080 nM T77365 C3SP8W 70693390 Ki = 1350 nM T77365 C8RS6V 70694477 Ki = 1000 nM T77365 C1KHZ2 70694510 Ki > 10000 nM T77365 CGW8U4 70695809 Ki = 3700 nM T77365 CL3E6M 70695810 Ki = 2450 nM T77365 CVU08A 70695812 Ki = 3950 nM T77365 C8XWN2 70696536 Ki = 125.89 nM T77365 C2EW3D 70696537 Ki = 1000 nM T77365 C7USK0 70696572 Ki >= 10000 nM T77365 CBN9A8 70697521 Ki = 96 nM T77365 C6HRB4 71077940 IC50 = 3480 nM T77365 C6NKY5 71078482 Ki = 9700 nM T77365 C50WGF 71078515 Ki = 4600 nM T77365 CFK50V 71110267 IC50 = 680 nM T77365 CS4T0U 71110270 Ki = 3500 nM T77365 C3ORQ5 71110347 IC50 = 1800 nM T77365 CAH09S 71110518 IC50 > 10000 nM T77365 C75JTG 71361867 Ki = 22600 nM T77365 CAR92Q 71364275 Ki > 10000 nM T77365 C31FGM 71412032 Ki = 20 nM T77365 CBZM95 71449068 Ki > 10000 nM T77365 CXZ40U 71450227 Ki = 1150 nM T77365 C38UKP 71450240 Ki = 29900 nM T77365 CXM83Y 71450241 Ki = 368 nM T77365 C9G0FP 71450242 Ki = 336 nM T77365 CC73UY 71450243 Ki = 279 nM T77365 C2PA9L 71450842 Ki = 100000 nM T77365 CTYM41 71450845 Ki = 5100 nM T77365 CW75JC 71450849 Ki = 6420 nM T77365 CPQ4Y9 71451659 Ki = 4110 nM T77365 C4LVT1 71452054 Ki = 352 nM T77365 CC2Q9H 71452055 Ki = 2730 nM T77365 CQ4CA3 71452056 Ki = 55.2 nM T77365 CWOB13 71452072 Ki = 446 nM T77365 CX52PV 71452672 Ki = 1300 nM T77365 CXF65C 71452801 Ki = 2700 nM T77365 C0NC4G 71453140 Ki = 1610 nM T77365 C9QD3W 71453871 Ki = 597 nM T77365 CKW2G6 71453872 Ki = 6430 nM T77365 C0VK4E 71453873 Ki = 132 nM T77365 CR8A0V 71453874 Ki = 91 nM T77365 CV0NW6 71453875 Ki = 245 nM T77365 C5S3FU 71453891 Ki = 155 nM T77365 C0M9CP 71453892 Ki = 208 nM T77365 CY1B4N 71453893 Ki = 3230 nM T77365 C76PJS 71453894 Ki = 233 nM T77365 CO02WB 71454439 Ki = 3800 nM T77365 C56VEI 71455599 Ki = 109 nM T77365 C79IVN 71455600 Ki = 407 nM T77365 CM2ZF9 71455601 Ki = 121 nM T77365 CEO64T 71455602 Ki = 1030 nM T77365 CPN0B7 71455603 Ki = 117 nM T77365 CUE71P 71455604 Ki = 177 nM T77365 CC1RD4 71455619 Ki = 92.5 nM T77365 C2ITP7 71455620 Ki = 147 nM T77365 CQ8U5S 71455621 Ki = 272 nM T77365 CB2E9C 71455622 Ki = 168 nM T77365 CTH1W7 71455623 Ki = 512 nM T77365 C1QLP9 71455624 Ki = 83.9 nM T77365 CVJZ12 71456194 Ki = 10000 nM T77365 CJBC05 71456195 Ki = 4800 nM T77365 CIE1Z5 71456490 Ki = 1800 nM T77365 C5BHA3 71457388 Ki = 251 nM T77365 CYTZ37 71457389 Ki = 185 nM T77365 C3H2QF 71457390 Ki = 38.2 nM T77365 CPBO67 71457391 Ki = 75.4 nM T77365 C12PEI 71457403 Ki = 157 nM T77365 C19MUP 71457404 Ki = 389 nM T77365 CS6Z4N 71457405 Ki = 248 nM T77365 C5RD0O 71457406 Ki = 701 nM T77365 C6MF5O 71457407 Ki = 130 nM T77365 CJA6M2 71457990 Ki = 10000 nM T77365 C5MR7O 71458343 Ki = 2000 nM T77365 CJO41A 71458816 Ki = 13.1 nM T77365 CU0YQ6 71459244 Ki = 900 nM T77365 CV3L0D 71459245 Ki = 1670 nM T77365 CDW92B 71459246 Ki = 1380 nM T77365 C5WX8S 71459247 Ki = 1080 nM T77365 CN79LY 71459248 Ki > 30000 nM T77365 C82QUK 71459249 Ki = 848 nM T77365 CC9I6G 71459250 Ki = 64.1 nM T77365 CQ7BP5 71459268 Ki = 77 nM T77365 CG8MI3 71459899 Ki = 3700 nM T77365 C8AY0D 71460344 Ki = 1610 nM T77365 CB9A8S 71461026 Ki = 124 nM T77365 C60OEP 71461027 Ki = 7490 nM T77365 CUDN57 71461028 Ki = 87.5 nM T77365 CJ9K0H 71461029 Ki = 593 nM T77365 CDX9O4 71461045 Ki > 30000 nM T77365 COU59X 71461116 Ki = 2370 nM T77365 CQ7V9L 71461900 Ki = 5000 nM T77365 CA0EJ2 71462751 Ki = 7690 nM T77365 CK7OB3 71462752 Ki = 136 nM T77365 CP07FL 71462753 Ki = 207 nM T77365 CK97MP 71462754 Ki = 798 nM T77365 CV1QN8 71462755 Ki = 46.1 nM T77365 COU6E4 71462772 Ki = 6120 nM T77365 CGC23V 71462773 Ki = 244 nM T77365 C1HAS6 71462774 Ki = 113 nM T77365 CHT04N 71462775 Ki = 814 nM T77365 C1N5MY 71464785 Ki > 1000 nM T77365 CGT9W5 71508481 Ki = 80 nM T77365 CCJN86 71511630 Ki = 100 nM T77365 CNKZ09 71528098 Ki > 60000 nM T77365 CZXY43 71561477 Ki > 10000 nM T77365 C0FJ1X 71561478 Ki > 10000 nM T77365 CYZE35 71561479 Ki > 10000 nM T77365 C3QJ5M 71561480 Ki > 10000 nM T77365 C65OJL 71561481 Ki > 10000 nM T77365 CF4T7N 71561482 Ki > 10000 nM T77365 C13TRN 71561483 Ki > 10000 nM T77365 C43UWM 71561593 Ki > 10000 nM T77365 C7CFR4 71561594 Ki > 10000 nM T77365 C4YZ8I 71561595 Ki > 10000 nM T77365 CYM5Q0 71561596 Ki > 10000 nM T77365 C6XV7D 71562554 Ki > 1000 nM T77365 CU8QC4 71562555 Ki > 10000 nM T77365 C2GOS6 71562556 Ki > 10000 nM T77365 CH7A3C 71562557 Ki > 1000 nM T77365 CI5JP8 71562669 Ki > 10000 nM T77365 CN25AT 71562670 Ki > 10000 nM T77365 CZG10K 71562924 Ki > 10000 nM T77365 C1RQ0X 71562925 Ki > 1000 nM T77365 CJ5M2B 71562926 Ki > 1000 nM T77365 CH45VQ 71562928 Ki = 430 nM T77365 C3XTO4 71562929 Ki = 390.5 nM T77365 C1SYX5 71563047 Ki > 10000 nM T77365 CX40FP 71563048 Ki = 423.4 nM T77365 C2A9VU 71563049 Ki = 260 nM T77365 CHVB51 71563050 Ki = 530.6 nM T77365 C4N2XD 71563051 Ki = 246.6 nM T77365 CL60DA 71563052 Ki = 306.9 nM T77365 C41JWM 71563053 Ki > 10000 nM T77365 CBD60O 71563170 Ki > 10000 nM T77365 C9PEA5 71563171 Ki = 467.3 nM T77365 CI74VT 71563173 Ki = 886.8 nM T77365 C5H3ZN 71563174 Ki > 10000 nM T77365 C3UD6V 71563175 Ki > 10000 nM T77365 C4DE7M 71563176 Ki = 93.9 nM T77365 C64RSC 71563296 Ki > 1000 nM T77365 C5DZM0 71563297 Ki > 1000 nM T77365 CSVQ36 71563298 Ki > 10000 nM T77365 C2Z9RH 71563299 Ki > 1000 nM T77365 C65EVL 71563300 Ki > 10000 nM T77365 CQ2SL9 71563301 Ki = 1144 nM T77365 C0PI4G 71563302 Ki > 10000 nM T77365 CT29GM 71570217 Ki = 49.4 nM T77365 CKGR23 71570366 Ki = 375.1 nM T77365 C6SU2O 71572050 IC50 = 1200 nM T77365 C14BCP 71572051 IC50 = 970 nM T77365 CB1YS4 71572385 IC50 = 490 nM T77365 CR0KX9 71572386 IC50 = 430 nM T77365 CI39JB 71601630 Ki = 246 nM T77365 C9J4OB 71601631 Ki = 325 nM T77365 CRQP84 71601632 Ki = 110 nM T77365 CN2BP6 71602912 Ki = 67.3 nM T77365 C76WQP 71602913 Ki = 3.7 nM T77365 C3J1QE 71602914 Ki = 683 nM T77365 CF4XL2 71602915 Ki = 4.7 nM T77365 CXD5L1 71602961 Ki = 9.7 nM T77365 CT4FI9 71603017 Ki = 207 nM T77365 C8UJ5P 71603087 Ki = 7.3 nM T77365 CER07O 71603088 Ki = 594 nM T77365 C0TOS6 71603089 Ki = 67.3 nM T77365 C09TYA 71603090 Ki = 173 nM T77365 CM87NU 71623050 Ki = 73 nM T77365 CYO2C8 71624864 IC50 = 182 nM T77365 C3T0UN 71624865 IC50 = 2630 nM T77365 CNU23Y 71624866 IC50 = 9770 nM T77365 CBP36E 71624867 IC50 = 54954.09 nM T77365 C2G5EP 71624868 IC50 > 100000 nM T77365 CL9I8T 71624992 IC50 = 4365.16 nM T77365 C7NSA1 71625116 IC50 = 10964.78 nM T77365 CP3ZX1 71625117 IC50 > 100000 nM T77365 CFW5O6 71625118 IC50 = 50.12 nM T77365 CF6C1L 71625119 IC50 > 10000 nM T77365 CMXC26 71625251 IC50 > 100000 nM T77365 CP64TE 71625252 IC50 = 38.9 nM T77365 CF31GC 71625253 IC50 = 181.97 nM T77365 C28ANX 71625254 IC50 = 9120 nM T77365 CV80KS 71625255 IC50 = 9770 nM T77365 CNZ17D 71657835 EC50 = 2290.87 nM T77365 CI0GU8 71660496 IC50 > 48500 nM T77365 C0YW1C 71680730 Ki = 62.4 nM T77365 CG6EY1 71680731 Ki > 1000 nM T77365 CN0WU1 71680732 Ki >= 1000 nM T77365 CK2Y6A 71680733 Ki = 39.5 nM T77365 CH5KU9 71680734 Ki = 115 nM T77365 CCM92I 71680890 Ki = 118 nM T77365 CS51FY 71680891 Ki = 91.8 nM T77365 C6HZ4O 71680894 Ki > 1000 nM T77365 CN0EZ6 71680895 Ki = 58.3 nM T77365 C30NCG 71681049 Ki = 44.3 nM T77365 C2TR7P 71681050 Ki > 10000 nM T77365 C2Y3KO 71681203 Ki = 82.5 nM T77365 C21UWV 71683091 Ki = 80.9 nM T77365 COWX82 71683092 Ki = 64.9 nM T77365 C3RD0E 71713167 Ki > 100000 nM T77365 C4BVA5 71717928 Ki = 140.8 nM T77365 CY9J0Z 71745501 Ki = 64 nM T77365 CS87DW 72164230 Ki = 10.98 nM T77365 C8GZ5E 72164231 Ki = 0.03 nM T77365 COR6T8 72164232 Ki = 0.027 nM T77365 CTWX78 72164233 Ki = 2.64 nM T77365 CAR8I1 72164234 Ki = 0.0047 nM T77365 CXZM13 72164235 Ki = 1.44 nM T77365 CL57OG 72164236 Ki = 54.8 nM T77365 CO1R8B 72164352 Ki = 9.6 nM T77365 C3H2GK 72164353 Ki = 0.14 nM T77365 C4REK7 72164354 Ki = 0.01 nM T77365 CHQ6M0 72164355 Ki = 1.8 nM T77365 CYN8X6 72164356 Ki = 7.61 nM T77365 CLFV53 72164357 Ki = 0.067 nM T77365 C9F1AX 72164358 Ki = 0.0042 nM T77365 CZ0G2X 72165213 Ki = 6100 nM T77365 C5EMX3 72197342 Ki = 128 nM T77365 C4E0QC 72197343 Ki > 10000 nM T77365 C76ASV 72197513 Ki = 562 nM T77365 CZW4Y0 72197514 Ki = 327 nM T77365 CUL8V0 72197515 Ki > 30000 nM T77365 CXF4U1 72197516 Ki > 30000 nM T77365 C3QYT8 72197517 Ki = 4870 nM T77365 C4W8LQ 72197698 Ki > 10000 nM T77365 CY8GU4 72197699 Ki > 10000 nM T77365 C6BUC3 72197700 Ki > 10000 nM T77365 C48QTY 72197701 Ki = 74.7 nM T77365 C4D8WO 72197702 Ki = 552 nM T77365 CAY6J2 72197703 Ki = 193 nM T77365 C6RDT4 72197880 Ki = 6.65 nM T77365 C7XN0S 72197881 Ki = 5950 nM T77365 C5J9QH 72197882 Ki = 14400 nM T77365 CB05ET 72197883 Ki = 179 nM T77365 C52QMK 72197884 Ki > 100000 nM T77365 CGY90F 72546539 Ki = 602.4 nM T77365 CWH6T3 72548703 IC50 = 9.2 nM T77365 CS81LQ 72696144 Ki = 4610 nM T77365 C1E4ZD 72696146 Ki = 3780 nM T77365 CQ35NL 72696147 Ki = 1350 nM T77365 CRN4B1 72696148 Ki = 5250 nM T77365 CWG0U4 72697647 Ki = 2120 nM T77365 CPB7K4 72697649 Ki = 284 nM T77365 CA5BI1 72697652 Ki = 253 nM T77365 C50SYX 72697785 Ki = 417 nM T77365 CXPB58 72697786 Ki = 322 nM T77365 CY1I8G 72697789 Ki = 626 nM T77365 CXDT98 72697790 Ki = 1200 nM T77365 CS7VK8 72697791 Ki = 346 nM T77365 CX69MI 72697928 Ki = 508 nM T77365 CEWO96 72697930 Ki = 317 nM T77365 CNP9S3 72697931 Ki = 231 nM T77365 C3NR4V 72697932 Ki = 311 nM T77365 CQ4IE7 72697933 Ki = 1110 nM T77365 CY94KO 72697934 Ki = 510 nM T77365 CO5K1Y 72698079 Ki = 628 nM T77365 CH6Z2U 72698223 Ki = 2530 nM T77365 CJ6IY1 72793900 Ki = 1.1 nM T77365 CR8YJ1 72945114 Ki = 24 nM T77365 C5OQ3F 72945115 Ki = 45 nM T77365 CZOX96 72945117 Ki = 9.5 nM T77365 CRFW68 72945315 Ki = 65 nM T77365 CM6P9F 72945317 Ki = 66 nM T77365 C8U2GW 72945318 Ki = 52 nM T77365 CR7M6U 72945319 Ki = 9.2 nM T77365 CR2GM4 72945321 Ki = 43 nM T77365 CW83DK 73213196 Ki > 10000 nM T77365 CRO2K8 73345315 Ki = 430 nM T77365 CRW73S 73345316 Ki > 10000 nM T77365 C5AB9Z 73346835 Ki = 480 nM T77365 CF1JN5 73347573 Ki > 10000 nM T77365 CM5B9S 73347862 Ki > 10000 nM T77365 CTJ0U3 73348946 Ki = 2010 nM T77365 CC3Y7G 73348947 Ki = 27 nM T77365 C2PTH6 73349106 Ki = 933.25 nM T77365 CI65VU 73349920 Ki = 1600 nM T77365 C4C0GK 73349930 Ki = 1300 nM T77365 CY5K9T 73350674 Ki = 6165.95 nM T77365 CHLF98 73350966 Ki > 10000 nM T77365 CE2YB8 73350967 Ki > 10000 nM T77365 CQSX70 73350968 Ki > 10000 nM T77365 C5YXO4 73352175 Ki = 6760.83 nM T77365 C5H8SI 73352180 Ki = 2511.89 nM T77365 CIH36P 73352882 Ki = 800 nM T77365 C35XEH 73352883 Ki = 850 nM T77365 C2M8PJ 73353634 Ki = 6165.95 nM T77365 C2IG8X 73353638 Ki = 467.74 nM T77365 CW18JX 73355444 Ki > 10000 nM T77365 C4HX2J 73355960 Ki = 1100 nM T77365 CH6G8N 73356702 Ki = 1778.28 nM T77365 CF8P0A 73356703 Ki = 6025.6 nM T77365 C86NPK 76308484 Ki = 16000 nM T77365 CMS65T 76309882 Ki = 59 nM T77365 CB84HP 76309883 Ki = 106 nM T77365 C02EBL 76309925 Ki = 1400 nM T77365 CX1H6Y 76310493 Ki = 3300 nM T77365 C9DL1B 76310832 Ki = 0.2 nM T77365 CGPZ23 76310922 Ki = 2530 nM T77365 CP9N0W 76311193 Ki = 25.12 nM T77365 CCX8V6 76311194 EC50 = 251.19 nM T77365 CQLE57 76311197 EC50 > 10000 nM T77365 CSV43U 76313599 Ki = 1270 nM T77365 CP2TA1 76313600 Ki = 50 nM T77365 CQ5Z4P 76313639 Ki = 333 nM T77365 CY8D4J 76313640 Ki > 100000 nM T77365 CB0WN9 76313641 Ki > 100000 nM T77365 C1C3LK 76314155 Ki = 2060 nM T77365 C25LDC 76314450 Ki = 0.4 nM T77365 CEO9I0 76314563 Ki = 2200 nM T77365 CZX45G 76314797 EC50 = 3981.07 nM T77365 C21BCT 76317721 Ki = 25600 nM T77365 C2K6XR 76317722 Ki = 2700 nM T77365 CY3V7H 76317723 Ki > 100000 nM T77365 CXQY23 76317724 Ki = 29900 nM T77365 CCY8V2 76318040 Ki = 0.29 nM T77365 CX3H8W 76318139 Ki = 2860 nM T77365 CL4JH8 76318403 EC50 = 2511.89 nM T77365 C9O4CQ 76320863 Ki = 2060 nM T77365 CKLB89 76320909 Ki = 980 nM T77365 CL46PW 76321429 Ki = 1600 nM T77365 CWO42D 76321430 Ki = 2100 nM T77365 CFN3M9 76321431 Ki = 23600 nM T77365 CY5TN2 76321753 Ki = 0.25 nM T77365 C4TO0S 76321824 Ki = 7490 nM T77365 CHCM51 76321825 Ki = 3150 nM T77365 C5R6OT 76322076 EC50 = 794.33 nM T77365 CK5Z6L 76324475 Ki = 57 nM T77365 CHWO53 76324476 Ki = 7.5 nM T77365 C3CE4B 76324522 Ki = 9090 nM T77365 C6AV9Z 76325026 Ki = 800 nM T77365 C1JV7S 76325027 Ki = 8600 nM T77365 CQ51JN 76325369 Ki = 0.31 nM T77365 C2DPT3 76325370 Ki = 0.045 nM T77365 CP4CY1 76325371 Ki = 0.042 nM T77365 C5J4ML 76325372 Ki = 8.09 nM T77365 COD78V 76325693 EC50 = 5011.87 nM T77365 C3FE0S 76325694 EC50 = 794.33 nM T77365 CC67KO 76328082 Ki > 100000 nM T77365 CA0MJ2 76328083 Ki = 8390 nM T77365 C72UFI 76328084 Ki = 11200 nM T77365 CNM0E1 76328596 Ki = 20500 nM T77365 CXTN91 76328597 Ki = 12000 nM T77365 C3TH4J 76328598 Ki = 3100 nM T77365 CQI9X5 76328599 Ki = 16400 nM T77365 C0AE9L 76328600 Ki > 100000 nM T77365 C5B0UO 76328910 Ki = 0.12 nM T77365 C5VEJ9 76328911 Ki > 10 nM T77365 C7K3AS 76329262 Ki = 79.43 nM T77365 C8O5KF 76329263 EC50 = 79.43 nM T77365 C9O0UH 76329264 EC50 = 501.19 nM T77365 CF82DA 76329265 EC50 = 1258.93 nM T77365 CPVN52 76329266 EC50 = 3162.28 nM T77365 C0E9DN 76330242 Ki = 7000 nM T77365 CG30CO 76331702 Ki = 18 nM T77365 C6QY2P 76331703 Ki = 89 nM T77365 CFNG34 76331754 Ki = 980 nM T77365 CMR14L 76331755 Ki = 2210 nM T77365 CQT81A 76332277 Ki = 3700 nM T77365 CH64XC 76332278 Ki = 4600 nM T77365 CQWD47 76332279 Ki > 100000 nM T77365 CJKD34 76332280 Ki = 9900 nM T77365 C1GZ8R 76332281 Ki = 17500 nM T77365 CVT1E3 76332599 Ki > 10 nM T77365 CVS3F8 76332600 Ki = 3.17 nM T77365 CIF6V7 76332686 Ki = 1760 nM T77365 CZ27KW 76332687 Ki = 3310 nM T77365 CYK39X 76332918 EC50 > 10000 nM T77365 C4S8NF 76332919 EC50 > 10000 nM T77365 CF68KC 76335303 Ki = 15 nM T77365 CL83MV 76335304 Ki = 110 nM T77365 C7KY5A 76335305 Ki = 33 nM T77365 CC5IO4 76335344 Ki = 2690 nM T77365 C7FE5D 76335345 Ki = 1270 nM T77365 CIT36F 76335346 Ki = 13200 nM T77365 CV05FX 76335917 Ki = 4100 nM T77365 CLN8S6 76335918 Ki = 24200 nM T77365 CM0D3G 76335919 Ki = 1100 nM T77365 CO86UR 76335920 Ki = 3500 nM T77365 CESR09 76335921 Ki = 2200 nM T77365 CR85PG 76335922 Ki = 5400 nM T77365 C3HE2N 76335923 Ki = 4700 nM T77365 C5DSC0 76335924 Ki > 100000 nM T77365 C5VM4Q 76336198 Ki = 0.072 nM T77365 C01BQD 76336523 Ki = 1584.89 nM T77365 C4Z3JY 76336524 Ki = 316.23 nM T77365 CH9WJ4 76336525 EC50 > 10000 nM T77365 CNL62P 76336526 EC50 > 10000 nM T77365 C5ZRE9 76336527 EC50 = 398.11 nM T77365 CI4M9P 85706712 Ki = 25500 nM T77365 CU5NE8 86302363 Ki = 3.8 nM T77365 CQS7X2 88448936 Ki = 4.1 nM T77365 CNZ2I8 89584875 IC50 = 450 nM T77365 C6PQW3 89819336 Ki = 0.6 nM T77365 CIS39L 89819339 Ki = 2 nM T77365 C0M7NI 90268057 Ki = 5.5 nM T77365 CY5P6I 90268061 Ki = 10.1 nM T77365 CE50JT 90655901 Ki = 4 nM T77365 CA4H1M 90665174 Ki = 4.1 nM T77365 CXK5T1 90665312 Ki = 1070 nM T77365 CWPT08 90665313 Ki > 10000 nM T77365 CM78DN 90665314 Ki > 10000 nM T77365 C8DRF0 90665315 Ki > 10000 nM T77365 CJIO86 90665316 Ki > 10000 nM T77365 C02JAH 90665317 Ki = 3760 nM T77365 C2K1SF 90665318 Ki = 2250 nM T77365 CH6KA8 90668272 Ki = 27.6 nM T77365 CX9E1Z 90668273 Ki = 9.2 nM T77365 CYR6N5 90668274 Ki = 7.2 nM T77365 C73XJB 90668275 Ki = 240 nM T77365 CFA6R0 90668276 Ki = 240 nM T77365 CC1KY8 90668277 Ki = 995 nM T77365 CU58ZA 91864603 Ki = 0.4 nM T77365 C0ROS7 101874280 Ki = 104 nM T77365 CPRH91 110171405 Ki = 300 nM T77365 CQI36D 117137080 Ki > 10000 nM T77365 CGBO72 118016229 IC50 = 820 nM T77365 CB74NK 118707149 Ki = 2530 nM T77365 C7UOD9 118707151 Ki = 1200 nM T77365 CFH85E 118707843 Ki = 65.2 nM T77365 COX73K 118707844 Ki = 11.1 nM T77365 CR13GS 118707845 Ki = 5.76 nM T77365 CS0WC2 118707846 Ki = 1520 nM T77365 C2A3FW 118707847 Ki = 12.4 nM T77365 CJ58XH 118707848 Ki = 51.4 nM T77365 CF78CL 118707849 Ki = 773 nM T77365 C3K7UV 118707850 Ki = 28.1 nM T77365 C0UFO4 118707851 Ki = 4.82 nM T77365 CSW70B 118707852 Ki = 183 nM T77365 CU9OE7 118707853 Ki = 42700 nM T77365 CGJW82 118707854 Ki = 24700 nM T77365 CUR32J 118707855 Ki = 50.3 nM T77365 C6O0RY 118707856 Ki = 50.1 nM T77365 CG10IH 118707857 Ki = 103 nM T77365 C9OHF2 118707858 Ki = 215 nM T77365 CW72CL 118707859 Ki = 37.4 nM T77365 CL0U3C 118707860 Ki = 43.4 nM T77365 CL3NG5 118707861 Ki = 121 nM T77365 C9BSD0 118707862 Ki = 32 nM T77365 CDTJ73 118707863 Ki = 122 nM T77365 CRDU39 118707864 Ki = 142 nM T77365 C6Y5VQ 118707865 Ki = 39.3 nM T77365 CBO8V9 118707866 Ki = 73.2 nM T77365 C4CU6D 118707867 Ki = 209 nM T77365 C4P5GH 118707868 Ki = 187 nM T77365 C9FKE5 118707869 Ki = 385 nM T77365 CNJ3Z4 118707870 Ki = 28.9 nM T77365 CXQY36 118707871 Ki = 235 nM T77365 C7SL4C 118707872 Ki = 351 nM T77365 CFR3Z1 118707873 Ki = 10200 nM T77365 C87ATB 118707874 Ki = 8180 nM T77365 C7HS6T 118707875 Ki = 6480 nM T77365 CXHQ82 118707876 Ki = 17600 nM T77365 CEQP75 118707877 Ki = 58.9 nM T77365 CY8OV1 118707878 Ki > 100000 nM T77365 CH5B6Y 118707879 Ki = 44.4 nM T77365 C3OJW0 118707880 Ki = 210 nM T77365 CM5BE7 118707881 Ki > 100000 nM T77365 CHR1E9 118707882 Ki = 3680 nM T77365 CZW6U4 118707883 Ki = 26900 nM T77365 COR57B 118707884 Ki = 7660 nM T77365 C8C9TQ 118707885 Ki = 33800 nM T77365 C0NQ2O 118707886 Ki = 596 nM T77365 CG68RH 118707887 Ki = 37300 nM T77365 C9CY3P 118707888 Ki = 33900 nM T77365 CNC81J 118707889 Ki = 3660 nM T77365 CM53PE 118707890 Ki = 1190 nM T77365 CL4B7K 118707891 Ki = 12400 nM T77365 CR20MO 118707892 Ki = 6390 nM T77365 C8WQ5E 118707893 Ki > 100000 nM T77365 CI6O9D 118707894 Ki = 18000 nM T77365 C28ABD 118707895 Ki > 100000 nM T77365 C56KNQ 118707896 Ki > 100000 nM T77365 C7LNI5 118708213 Ki = 89 nM T77365 C74OYF 118708214 Ki = 410 nM T77365 CBG4I3 118708219 Ki = 213 nM T77365 CFOC02 118708225 Ki = 154 nM T77365 C50PKS 118708228 Ki = 521 nM T77365 CWU94Y 118708234 Ki = 55 nM T77365 CI29WS 118708235 Ki = 153 nM T77365 C2B0KW 118708236 Ki = 147 nM T77365 C0MXW8 118708237 Ki = 790 nM T77365 CX2B8P 118708238 Ki = 102 nM T77365 CQWJ06 118708239 Ki = 146 nM T77365 CL6P0G 118708240 Ki = 722 nM T77365 CYO73E 118714540 EC50 = 5.86 nM T77365 CJEW03 118714541 Ki = 4360 nM T77365 C0N4FO 118714542 Ki = 3280 nM T77365 CQZ6I2 118714543 Ki = 267 nM T77365 CI76CX 118719026 Ki = 6.4 nM T77365 CN4SK2 118721485 Ki = 2401 nM T77365 CQ0AD4 118723498 Ki = 51 nM T77365 CO3JQ2 118723499 Ki = 2595.4 nM T77365 CD1W6R 118723501 Ki = 69.2 nM T77365 C1SN3J 118723507 Ki = 75.5 nM T77365 C8YUA2 118723508 Ki = 662.4 nM T77365 CC94IX 118725995 IC50 = 35 nM T77365 CL1I3E 118725996 IC50 > 100000 nM T77365 C3AU5G 118725997 IC50 = 63 nM T77365 C5EVX3 118726000 IC50 = 109.65 nM T77365 CAM4W1 118726001 IC50 = 40.74 nM T77365 C7MVA4 118726004 IC50 = 436.52 nM T77365 CP8YI2 118726005 IC50 = 134.9 nM T77365 C5SIX4 118726006 IC50 = 120.23 nM T77365 C6MV1Y 118726008 IC50 = 32 nM T77365 CH5W0A 118726009 IC50 = 1122.02 nM T77365 CWN6M4 118726010 IC50 = 912 nM T77365 CM7NZ9 118726011 IC50 = 1778 nM T77365 C65OZV 118726012 IC50 = 1737.8 nM T77365 CZ3C8H 118726013 IC50 = 8511 nM T77365 C0OUK6 118726016 IC50 = 1514 nM T77365 CK1S2U 118726021 IC50 = 58.88 nM T77365 CVQ9X3 118728358 Ki > 6000 nM T77365 C5Z4TW 118728359 Ki = 730 nM T77365 CHSP62 118728360 Ki = 300 nM T77365 C8HVS9 118728362 Ki = 1100 nM T77365 C7GSL5 118728364 Ki = 6600 nM T77365 C9BFI0 118728365 Ki > 2100 nM T77365 CBJ36S 118728367 Ki = 830 nM T77365 C9H5SR 118728368 Ki = 240 nM T77365 C7LUH2 118728369 Ki = 130 nM T77365 CB2X4E 118729221 Ki = 110 nM T77365 C6RXB2 118729222 Ki = 110 nM T77365 C2NBS8 118729966 Ki = 6450 nM T77365 CBH8G1 118729967 Ki > 30000 nM T77365 CA3IK7 118729968 Ki > 30000 nM T77365 CTL02Y 118729969 Ki > 10000 nM T77365 CGTA19 118729970 Ki = 28400 nM T77365 C8KX7U 118729971 Ki = 18000 nM T77365 CWJ48N 118729972 Ki > 100000 nM T77365 CU0W7P 118729973 Ki > 30000 nM T77365 CAS85G 118729974 Ki > 10000 nM T77365 CFX4R9 118729975 Ki = 22300 nM T77365 C6VC5A 118729976 Ki = 3440 nM T77365 CNG5S7 118729977 Ki > 10000 nM T77365 CD6GZ2 118729978 Ki > 30000 nM T77365 C03XWO 118729979 Ki > 10000 nM T77365 CZD98F 118729980 Ki = 5670 nM T77365 CE5Z7R 118729981 Ki = 9660 nM T77365 CBV0J4 118729982 Ki > 30000 nM T77365 C2A5CU 118729983 Ki = 26600 nM T77365 CM3S0N 118732278 Ki = 3000 nM T77365 CWQ54J 118732279 Ki = 9200 nM T77365 CQL0K7 118732280 Ki > 80000 nM T77365 CRK7H9 118732281 Ki = 15700 nM T77365 CK24DH 118732282 Ki = 2000 nM T77365 CP78KH 118732283 Ki = 2600 nM T77365 CEO92J 118732284 Ki = 5000 nM T77365 CJ6YF9 118732285 Ki = 4800 nM T77365 CW62JS 118732286 Ki = 16100 nM T77365 CXW9U6 118732287 Ki = 11500 nM T77365 C06FRT 118732288 Ki > 100000 nM T77365 CR2CO8 118732289 Ki = 11800 nM T77365 C94GHE 118732290 Ki = 3300 nM T77365 COJ86X 118732291 Ki = 2800 nM T77365 C1KDT4 118732292 Ki > 100000 nM T77365 C7BO1N 118732293 Ki = 2300 nM T77365 C4EFY5 118732294 Ki = 5700 nM T77365 CKV50L 118732295 Ki = 3700 nM T77365 CT3Q9E 118732296 Ki = 6100 nM T77365 CLRK73 118732297 Ki = 7500 nM T77365 CE85HO 118732298 Ki = 6000 nM T77365 C9Y6EK 118732299 Ki = 4200 nM T77365 CNJ1H0 118732300 Ki > 100000 nM T77365 CX6IN3 118732301 Ki > 100000 nM T77365 C4N6ZT 118732302 Ki > 100000 nM T77365 CDAZ14 118732303 Ki > 100000 nM T77365 CZ7TM6 118732304 Ki > 100000 nM T77365 CXZW46 118732305 Ki > 100000 nM T77365 CWX3P4 118732306 Ki = 7300 nM T77365 CXRT76 118732307 Ki = 8800 nM T77365 CK0NS3 118732308 Ki = 5700 nM T77365 CRFJ71 118732309 Ki = 2400 nM T77365 CT90VA 118732971 EC50 = 2.36 nM T77365 CXM53U 118732972 Ki = 778 nM T77365 CF4G3P 118732973 EC50 = 238 nM T77365 C3E2BJ 118732974 EC50 = 9.75 nM T77365 C1U2FS 118732975 EC50 = 5.31 nM T77365 C4YS5J 118732976 EC50 = 7.71 nM T77365 CZ7QU0 118732977 EC50 = 12.8 nM T77365 CHP93T 118732978 EC50 = 25.1 nM T77365 CBT95M 118732979 EC50 = 33.2 nM T77365 CZ3X0P 118732980 EC50 = 8.4 nM T77365 CMDH59 118732981 EC50 = 28.8 nM T77365 C7MZ9V 118732982 EC50 = 9.04 nM T77365 CVS8R0 118734340 Ki = 55 nM T77365 C91DBT 118734341 Ki = 237 nM T77365 CV1JE8 118734342 Ki = 659 nM T77365 C8AB7F 118734343 Ki = 967 nM T77365 CLWV70 118734344 Ki = 98 nM T77365 CP7SE9 118734345 Ki = 25 nM T77365 CC0RE9 118734346 Ki = 29 nM T77365 CV6X3F 118734347 Ki = 92 nM T77365 CN8RI9 118734348 Ki = 36 nM T77365 CEZ86B 118734349 Ki = 24 nM T77365 C1QPJ3 118734350 Ki = 88 nM T77365 CFH92R 118734351 Ki = 43 nM T77365 CR8FT9 118734352 Ki = 56 nM T77365 C8Y7QW 118734353 Ki = 30 nM T77365 CR3Y1J 118734354 Ki = 84 nM T77365 C5DL3X 118734355 Ki = 23 nM T77365 CYB49C 118734356 Ki = 72 nM T77365 CZE09N 118734357 Ki = 7.76 nM T77365 CB7J1G 118734358 Ki = 18.21 nM T77365 C79RHZ 118734359 Ki = 95 nM T77365 CSAH95 118734360 Ki = 277 nM T77365 C1CBG3 118734361 Ki = 34 nM T77365 CN9S1Y 118734362 Ki = 26 nM T77365 C5SQA1 118734363 Ki = 33 nM T77365 CDVO89 118734364 Ki = 5.48 nM T77365 CQ73IF 118734365 Ki = 4.78 nM T77365 C43VAO 118734366 Ki = 24 nM T77365 C4NQV6 118734367 Ki > 10000 nM T77365 CGF84C 118734368 Ki > 10000 nM T77365 C94UXF 118734369 Ki > 10000 nM T77365 CU0K8H 118734370 Ki = 682 nM T77365 CPY5O0 118734371 Ki = 745 nM T77365 CLI1V7 118734372 Ki = 33 nM T77365 CX08QC 118734373 Ki = 235 nM T77365 CD3BV5 118734374 Ki = 24 nM T77365 C58VBC 118734375 Ki > 10000 nM T77365 C0U1NA 118734376 Ki = 16.32 nM T77365 CZH87J 118734377 Ki = 52 nM T77365 C7OW4T 121225598 Ki = 31 nM T77365 C6R5EX 122178744 Ki > 1000 nM T77365 CH7X6K 122178745 Ki > 1000 nM T77365 C4EW6R 122178746 Ki > 1000 nM T77365 C0ORM6 122178747 Ki > 1000 nM T77365 C7WCK3 122178748 Ki > 1000 nM T77365 C0V6CM 122178749 Ki > 1000 nM T77365 C6CQP9 122178750 Ki > 1000 nM T77365 C3Z2FP 122178751 Ki > 1000 nM T77365 C1HA2V 122178752 Ki > 1000 nM T77365 C4LN2B 122178753 Ki > 1000 nM T77365 CC6X3Q 122178754 Ki > 1000 nM T77365 CA25IQ 122178755 Ki > 1000 nM T77365 CSKN51 122178756 Ki > 1000 nM T77365 C79XUV 122178757 Ki > 1000 nM T77365 C1MA9K 122182829 Ki = 8.6 nM T77365 C06YKW 122182830 Ki = 5.3 nM T77365 CT6L2Q 122182831 Ki = 13.3 nM T77365 CZ45UW 122182832 Ki = 37.5 nM T77365 CA1I5D 122182833 Ki = 39.9 nM T77365 C9S2AG 122182834 Ki = 92.9 nM T77365 C2R5TF 122182835 Ki = 26.5 nM T77365 CQI46V 122182836 Ki = 8.9 nM T77365 CDQ50Z 122182837 Ki = 7.7 nM T77365 CU7NC1 122182838 Ki = 4.8 nM T77365 CGJ4S6 122182839 Ki = 24.6 nM T77365 CKR73I 122182840 Ki = 22.8 nM T77365 CE7M1W 122182841 Ki = 6.7 nM T77365 C8LIP2 122182842 Ki = 1.4 nM T77365 CWE9G8 122182843 Ki = 5.2 nM T77365 C6GTI8 122182881 Ki = 20 nM T77365 C0D4IR 122182882 Ki = 9.4 nM T77365 C6Y7TV 122444911 Ki = 0.5 nM T77365 C8TVD5 122444916 Ki = 0.2 nM T77365 CUQ03X 122444918 Ki = 9.6 nM T77365 CAOC96 122444919 Ki = 10 nM T77365 C7W1EU 122444920 Ki = 0.8 nM T77365 CE2O8R 122444921 Ki = 0.6 nM T77365 C4CA3G 122444930 Ki = 24 nM T77365 CW58PY 122444937 Ki = 160 nM T77365 C1G3QV 122444939 Ki = 3 nM T77365 CV9XW2 122444941 Ki = 7.7 nM T77365 CU2A5O 122444945 Ki = 0.2 nM T77365 C2WOJ7 122444955 Ki = 1.5 nM T77365 C95ULS 122444963 Ki = 0.2 nM T77365 CWXB61 122444964 Ki = 7.8 nM T77365 CU65EJ 122444974 Ki = 0.2 nM T77365 CL0SB8 122444975 Ki = 4.6 nM T77365 CG71FB 122444983 Ki = 180 nM T77365 CLW58S 122444984 Ki = 0.2 nM T77365 C8QZN9 122444991 Ki = 2.3 nM T77365 C5FMS9 122444992 Ki = 0.7 nM T77365 CIT59V 122444996 Ki = 0.5 nM T77365 CW4LR8 122445001 Ki = 86 nM T77365 C76ATO 122445003 Ki = 3 nM T77365 C9F7RX 122445009 Ki = 2 nM T77365 C7WIN8 122445018 Ki = 21.5 nM T77365 CB5C8V 122485306 Ki = 6.7 nM T77365 CNQJ76 122485307 Ki = 7.6 nM T77365 C5M2OL 122485308 Ki = 6.7 nM T77365 CJM03O 122485352 Ki = 0.4 nM T77365 CE1ZM8 122485358 Ki = 5 nM T77365 CU8HB2 123131614 Ki = 460 nM T77365 CX43WO 123131616 Ki = 1750 nM T77365 CKW26O 123131618 Ki = 920 nM T77365 C1C5XE 127025020 Ki = 0.5 nM T77365 CBQY40 127025021 Ki = 0.3 nM T77365 CT2AL0 127025022 Ki = 4.4 nM T77365 C02MLK 127025023 Ki = 3.1 nM T77365 C9OR6D 127025959 EC50 = 15848.93 nM T77365 CTL62C 127026187 Ki = 836 nM T77365 CXG31M 127026188 Ki = 1.1 nM T77365 C0MWD8 127026257 EC50 = 5754.4 nM T77365 CZ61LK 127034966 EC50 > 5011.87 nM T77365 CA0SN5 127034967 EC50 > 5011.87 nM T77365 CH6L8J 127035004 Ki = 115 nM T77365 C2BM4D 127035624 Ki = 86.9 nM T77365 CFJ95C 127035625 Ki = 7.87 nM T77365 CPY0S3 127035626 Ki = 1.44 nM T77365 CDWC03 127035803 Ki = 300 nM T77365 CH41BT 127035804 Ki = 393 nM T77365 C7AHR2 127035805 Ki = 23.6 nM T77365 C92RXW 127035806 Ki = 5.39 nM T77365 CGD59Y 127035832 Ki = 143 nM T77365 CX29PN 127035833 Ki = 397 nM T77365 C4Y3XI 127035834 Ki = 177 nM T77365 CJM9Z1 127036437 Ki = 49.3 nM T77365 CM63GQ 127036438 Ki = 99.6 nM T77365 C59HYJ 127036640 Ki = 113 nM T77365 CJ52XA 127036641 Ki = 560 nM T77365 CX9H5M 127036642 Ki = 905 nM T77365 C4F2WP 127036740 Ki = 194 nM T77365 C3QVM7 127036741 Ki = 2150 nM T77365 C3E7ZT 127036742 Ki = 1020 nM T77365 CGM30I 127036810 Ki = 15.2 nM T77365 CR7OT4 127036811 Ki = 173 nM T77365 CR58OX 127036812 Ki = 394 nM T77365 C65YKX 127036844 Ki = 20.4 nM T77365 CLCF05 127036845 Ki = 235 nM T77365 C5K3MR 127036846 Ki = 112 nM T77365 CB8HG0 127036933 Ki = 95.2 nM T77365 C1MS0C 127036976 Ki = 21.8 nM T77365 CQR43P 127036977 Ki = 43.6 nM T77365 C82FEM 127037758 Ki = 64000 nM T77365 C7LV5T 127038039 Ki = 3708 nM T77365 C64GTU 127038104 Ki > 200000 nM T77365 CB1IM0 127038106 Ki > 200000 nM T77365 C0VX6H 127038108 Ki = 35000 nM T77365 C72DGU 127038339 EC50 = 48 nM T77365 C2YT3C 127038355 Ki = 503 nM T77365 C3CMX4 127038356 Ki = 36 nM T77365 CB63LH 127038545 Ki = 126 nM T77365 C3RV0U 127038566 Ki = 25 nM T77365 CB5F1H 127038752 EC50 = 5.5 nM T77365 CR3A5Y 127038753 Ki = 13.2 nM T77365 C2KN6C 127038754 EC50 = 9.6 nM T77365 CN2R1H 127038755 EC50 = 10.6 nM T77365 C86CAO 127038756 Ki = 6.9 nM T77365 C5IL3Q 127038757 Ki = 10.3 nM T77365 CHV76Y 127038890 Ki = 26.7 nM T77365 CB76CP 127038901 Ki = 3.6 nM T77365 CQ7SD5 127038919 Ki = 1035 nM T77365 C4GA2B 127039480 Ki > 200000 nM T77365 C48TMH 127039482 Ki > 200000 nM T77365 CEV63D 127039484 Ki > 200000 nM T77365 CZ6X7P 127039486 Ki > 200000 nM T77365 CJ6IR0 127039488 Ki > 200000 nM T77365 C2OGT9 127040015 Ki = 10.1 nM T77365 CSU8G3 127040016 Ki = 20 nM T77365 C72WLA 127040044 Ki > 200000 nM T77365 CUD27T 127040064 Ki = 113 nM T77365 CL8SZ1 127040348 Ki = 1110 nM T77365 C7J1VL 127040399 Ki > 200000 nM T77365 CY4G8A 127040403 Ki = 12000 nM T77365 C9OG1N 127040410 Ki = 1180 nM T77365 CM5EQ3 127040561 Ki = 6.6 nM T77365 CA3HW8 127040562 Ki = 5.4 nM T77365 CVX0J9 127040563 Ki = 45 nM T77365 CNJ86G 127040564 Ki = 8.4 nM T77365 C51KHG 127040602 Ki > 10000 nM T77365 CRKD65 127040671 Ki = 2770 nM T77365 C64YFB 127041015 Ki = 3.1 nM T77365 C6G8HJ 127041016 Ki = 8.2 nM T77365 C3HEG8 127041017 Ki = 1.8 nM T77365 CWJ63T 127041018 Ki = 927 nM T77365 CNL13K 127041019 Ki = 15 nM T77365 CN8YI1 127041044 Ki = 2.7 nM T77365 CVA6S8 127041419 Ki = 16.4 nM T77365 CXA76Q 127041420 EC50 = 4.1 nM T77365 CN2R5C 127041421 Ki = 20.9 nM T77365 CK5ST2 127041635 Ki = 15.2 nM T77365 CI0BX5 127041636 Ki = 73.2 nM T77365 C15TGL 127041637 Ki = 245 nM T77365 CN5PD8 127041638 Ki = 1536 nM T77365 CN0J6D 127041683 Ki > 200000 nM T77365 C2KNY6 127041935 Ki = 12 nM T77365 C0F5YR 127041936 Ki = 6.9 nM T77365 CQ4HV3 127042140 Ki = 13.6 nM T77365 CEN1Z7 127042141 Ki = 14 nM T77365 CW93CB 127042203 Ki > 10000 nM T77365 CV31PY 127042204 Ki > 10000 nM T77365 C8D4GN 127042408 Ki = 1400 nM T77365 CA1XD7 127042409 Ki = 6.6 nM T77365 C29QAL 127042479 Ki = 160 nM T77365 CSR5P7 127042548 Ki > 10000 nM T77365 CXN90T 127042899 Ki = 4.4 nM T77365 CAZ71O 127042900 Ki = 4.8 nM T77365 C7ZOD5 127042993 Ki = 80 nM T77365 C10OFL 127042994 Ki = 547 nM T77365 CGE9O0 127042995 Ki = 13000 nM T77365 CCV4W8 127042996 Ki = 1020 nM T77365 C4JR2S 127042997 Ki = 181 nM T77365 CD23GH 127043299 Ki = 330 nM T77365 CG8F3I 127043648 Ki = 3260 nM T77365 CZ5BA7 127043662 Ki = 2180 nM T77365 C1J3PR 127043818 Ki = 245 nM T77365 C8V5EN 127043828 Ki = 546 nM T77365 CMJL86 127044142 Ki = 2260 nM T77365 CYS6Z4 127044283 Ki = 466 nM T77365 CC6MG4 127044514 Ki = 974 nM T77365 CW18JP 127044515 Ki = 313 nM T77365 C4O7WX 127044516 Ki = 3180 nM T77365 C3KQS4 127044517 Ki = 153 nM T77365 CE1A4H 127044518 Ki = 102 nM T77365 CQJ71U 127044681 Ki = 351 nM T77365 C7V4HX 127044785 Ki = 2960 nM T77365 CLXU52 127044795 Ki = 1110 nM T77365 C5FC3T 127044855 Ki = 200 nM T77365 C53KHG 127045164 Ki = 8110 nM T77365 C5LC0U 127045165 Ki = 1050 nM T77365 CGS9B5 127045166 Ki > 100000 nM T77365 C8NV5Y 127045167 Ki = 1030 nM T77365 C2R9PY 127045168 Ki = 1010 nM T77365 C0RMT7 127045169 Ki = 666 nM T77365 C7I3NV 127045170 Ki = 921 nM T77365 C6UK3Q 127045631 Ki = 2380 nM T77365 C8MT9L 127045699 Ki = 57 nM T77365 C02HYP 127045700 Ki = 51 nM T77365 C6VU1I 127045701 Ki = 6.21 nM T77365 C2GH3Q 127045815 Ki = 99 nM T77365 C4MQU2 127045909 Ki = 38 nM T77365 CQ1IB0 127045910 Ki = 14 nM T77365 CDHL50 127046050 Ki = 5.26 nM T77365 C80WYL 127046438 Ki = 412 nM T77365 CH8W3C 127046493 Ki = 5.37 nM T77365 COE1R5 127046494 Ki = 17 nM T77365 C72JQB 127046495 Ki = 9.23 nM T77365 C9OQ3P 127046496 Ki = 3.62 nM T77365 C51CEW 127047146 Ki = 518 nM T77365 C6WC1L 127047147 Ki = 147 nM T77365 C34CWL 127047737 Ki = 647 nM T77365 CBW49E 127047803 Ki = 240 nM T77365 C09DLO 127047851 Ki = 320 nM T77365 CC9U3O 127047927 Ki = 195 nM T77365 C5O9YM 127047928 Ki = 362 nM T77365 CV3K4L 127047929 Ki = 89 nM T77365 CNH42R 127051230 Ki = 9870 nM T77365 C97UBL 127051231 Ki > 100000 nM T77365 CQ3AL7 127051523 IC50 = 4400 nM T77365 C19MPD 127051839 IC50 = 5600 nM T77365 CU79JS 127051840 IC50 = 3400 nM T77365 CZ9NH5 127051849 Ki = 18800 nM T77365 C4A3IX 127051850 Ki > 100000 nM T77365 C8ACT1 127051851 Ki = 14700 nM T77365 CY2B7M 127051852 Ki = 20600 nM T77365 CPN29G 127052152 Ki > 100000 nM T77365 CB6R7Z 127052168 Ki = 7480 nM T77365 C2N7HC 127052751 IC50 = 8100 nM T77365 C1TJ7B 132578491 Ki = 230 nM T77365 C5CKG0 132578492 Ki = 595 nM T77365 CVS8H1 132578493 Ki = 203 nM T77365 CKIA45 132933622 Ki = 35700 nM T77365 CA31YG 132938348 Ki = 1080 nM T77365 C02UQE 132941757 Ki = 0.2 nM T77365 CJ54MF 132991405 IC50 = 0.0019 nM T77365 C75XIA 132991406 IC50 = 0.095 nM T77365 C9GE3Z 134132656 Ki = 1 nM T77365 C3UC1T 134132667 Ki = 17 nM T77365 C2I7AE 134132684 Ki = 18 nM T77365 CHSK61 134133787 Ki = 91 nM T77365 CH53WN 134134340 Ki = 2480 nM T77365 CZ8HL0 134134668 Ki = 1750 nM T77365 C6G4CW 134135745 Ki = 2200 nM T77365 C9A6KG 134138183 Ki = 1880 nM T77365 CR38DS 134138275 Ki = 20 nM T77365 C7WPX1 134138322 IC50 = 31 nM T77365 C8RVZ7 134138658 Ki = 4.7 nM T77365 CH0FX4 134138769 Ki = 3940 nM T77365 CV38YZ 134138961 IC50 = 123 nM T77365 CIAY28 134139825 Ki = 782 nM T77365 CBJW17 134140823 Ki = 154 nM T77365 C68AXD 134141831 Ki = 2200 nM T77365 C2KSZ9 134142435 Ki = 0.82 nM T77365 C06AXV 134142495 IC50 = 9 nM T77365 C5ZAD2 134142611 Ki = 16 nM T77365 CR1YQ6 134142843 Ki = 14000 nM T77365 CSUL60 134142882 Ki = 251 nM T77365 CXFG86 134143159 Ki = 1.3 nM T77365 C08RJA 134143536 Ki = 2690 nM T77365 C5L9BD 134143752 Ki = 1570 nM T77365 CWG9Q2 134144288 Ki = 7.2 nM T77365 C9T5ME 134147675 Ki = 36 nM T77365 C3L2PZ 134147788 IC50 = 18 nM T77365 CRA5O4 134147994 Ki = 58 nM T77365 C4MDF2 134148336 Ki = 1389 nM T77365 CPI01N 134149255 Ki = 30 nM T77365 CGT32F 134150875 Ki = 98 nM T77365 CGXA08 134151211 Ki = 65 nM T77365 CNET28 134151346 Ki = 17 nM T77365 C8PT9W 134152052 Ki = 4320 nM T77365 C73ISY 134152157 Ki = 2950 nM T77365 CA29KP 134152503 Ki = 129 nM T77365 C1JK6T 134152846 Ki = 40 nM T77365 CK7M8Y 134153079 Ki = 1.3 nM T77365 C7UOJ8 134156506 Ki = 1520 nM T77365 C48WTR 134156643 Ki = 120 nM T77365 C20RNA 134157761 Ki = 8.21 nM T77365 C1GY2T 135156251 EC50 > 10000 nM T77365 C08ZQW 135404340 Ki > 10000 nM T77365 CC0P2Z 135405211 IC50 = 2600 nM T77365 C9WD5K 135405767 Ki > 1000 nM T77365 C61NZE 135409562 Ki = 470 nM T77365 C2ATW9 135409793 Ki = 49 nM T77365 CRVK68 135409825 Ki = 1000 nM T77365 C5T2ZE 135409960 Ki > 1000 nM T77365 C6G0HA 135416050 Ki > 1000 nM T77365 CI0HT3 135416055 Ki > 1000 nM T77365 C1IEY0 135418256 IC50 > 10000 nM T77365 C0C5IU 135418454 Ki = 31 nM T77365 C0Z8RU 135421343 Ki > 1000 nM T77365 CW16MF 135421366 Ki > 1000 nM T77365 CUA67Z 135423046 Ki = 520 nM T77365 CLK7X1 135427226 IC50 = 550 nM T77365 CY9QI4 135428630 Ki = 1600 nM T77365 C7P2ME 135428645 Ki = 4400 nM T77365 C5OZ0L 135428653 Ki = 18000 nM T77365 CI4Z3R 135430228 Ki > 1000 nM T77365 CZA5F9 135436760 Ki > 1000 nM T77365 CJ6AW4 135437132 Ki = 88 nM T77365 CNJ9P7 135437142 IC50 = 3300 nM T77365 CB67JM 135437331 Ki = 8800 nM T77365 C6HN3Z 135438480 Ki = 532 nM T77365 CJT02K 135439354 Ki = 1778.28 nM T77365 C4Y9OF 135439478 Ki = 1300 nM T77365 CI4S7C 135440168 Ki > 1000 nM T77365 CR9W5J 135440414 Ki > 1000 nM T77365 C1UNH9 135440428 Ki > 1000 nM T77365 CXY13D 135440607 IC50 = 180 nM T77365 C3JA5S 135442119 Ki = 25 nM T77365 CAG0W3 135442266 IC50 = 900 nM T77365 C5YUC2 135443302 Ki > 1000 nM T77365 CO87CV 135443324 Ki > 1000 nM T77365 CWD8M7 135443353 Ki > 1000 nM T77365 C4KLO0 135443378 Ki > 1000 nM T77365 CAO3L2 135443744 IC50 = 510 nM T77365 CG9IK2 135444614 Ki = 49 nM T77365 CLK1W7 135445415 Ki = 3.467 nM T77365 CLY1V5 135447756 IC50 = 23 nM T77365 C9UCG0 135448286 Ki > 1000 nM T77365 C7D0AO 135450786 IC50 = 200 nM T77365 C0B1XV 135454766 Ki > 1000 nM T77365 C28AWC 135463688 Ki = 3500 nM T77365 C4DUN5 135464144 Ki = 892 nM T77365 C08VZH 135464239 Ki = 1200 nM T77365 C2Z0TJ 135465623 IC50 = 56 nM T77365 CK47BF 135465712 Ki = 25 nM T77365 CU14JT 135465774 Ki > 1000 nM T77365 C1F5CA 135465776 Ki > 1000 nM T77365 C04XNV 135465778 Ki > 1000 nM T77365 CBV8I2 135465784 Ki > 1000 nM T77365 C7E2CQ 135465796 Ki > 1000 nM T77365 CX04SI 135470376 IC50 = 47 nM T77365 C15FUA 135470377 IC50 = 58 nM T77365 C0YZ3B 135470411 Ki > 1000 nM T77365 C5F1TQ 135475602 IC50 = 360 nM T77365 CW4V3S 135475677 Ki = 25 nM T77365 CPQ3J6 135477916 Ki > 1000 nM T77365 CXJ12O 135479920 IC50 = 188 nM T77365 CK52RH 135483531 Ki > 1000 nM T77365 CTU21N 135483619 Ki > 1000 nM T77365 CJ91TZ 135484407 IC50 > 10000 nM T77365 C7A8ML 135484632 IC50 > 10000 nM T77365 CI8R0L 135485985 Ki = 20 nM T77365 CE26MK 135486084 Ki > 1000 nM T77365 CH0AR8 135486118 Ki > 1000 nM T77365 C94GIL 135490950 Ki = 24.3 nM T77365 CVG5M0 135493238 Ki > 1000 nM T77365 CCX3D7 135493268 Ki > 1000 nM T77365 CF06CK 135493272 Ki > 1000 nM T77365 CS3OC8 135493279 Ki > 1000 nM T77365 C9RS5H 135493280 Ki > 1000 nM T77365 CEI8W7 135493281 Ki > 1000 nM T77365 C25QGD 135493285 Ki > 1000 nM T77365 CN10IO 135493286 Ki > 1000 nM T77365 C7O1NS 135493290 Ki > 1000 nM T77365 CV4X0H 135493292 Ki > 1000 nM T77365 C5OK7A 135499926 Ki > 1000 nM T77365 CG3V6J 135501712 Ki = 45 nM T77365 CU8W5N 135508372 Ki > 1000 nM T77365 C28UOK 135509755 Ki = 980 nM T77365 CHM19U 135512719 IC50 = 46 nM T77365 C89IWT 135512738 IC50 = 210 nM T77365 CI03HR 135512751 IC50 = 7800 nM T77365 CSRL27 135512752 IC50 = 67 nM T77365 CTB6R7 135515408 IC50 > 10000 nM T77365 CFQ38U 135515507 Ki = 248 nM T77365 C9J5WF 135516512 IC50 = 2500 nM T77365 CCHU96 135516528 Ki = 25 nM T77365 C46YPU 135519330 Ki > 1000 nM T77365 CG64XS 135522362 Ki > 1000 nM T77365 C1E2ZK 135522363 Ki > 1000 nM T77365 C2CL8J 135522364 Ki > 1000 nM T77365 C2AHQ6 135522367 Ki > 1000 nM T77365 CF9XI7 135522375 Ki > 1000 nM T77365 C4NG7Y 135522388 Ki > 1000 nM T77365 C9A7QL 135522390 Ki > 1000 nM T77365 CUNG36 135522391 Ki > 1000 nM T77365 CFJ8P2 135525108 IC50 > 10000 nM T77365 C2WJI6 135529341 Ki > 1000 nM T77365 C7ARF8 135529362 Ki > 1000 nM T77365 C2V3CX 135529371 Ki > 1000 nM T77365 CVXF23 135529372 Ki > 1000 nM T77365 CJ86ZY 135529373 Ki > 1000 nM T77365 CESZ83 135529396 Ki > 1000 nM T77365 CJ4Y1H 135529398 Ki > 1000 nM T77365 C3V0NZ 135537639 IC50 = 120 nM T77365 C1OS2X 135542443 IC50 = 18 nM T77365 C8I2FM 135542466 Ki = 19 nM T77365 CU3F1O 135542558 Ki = 125 nM T77365 C51PIY 135543600 Ki = 572 nM T77365 CF3UQ4 135543624 Ki = 28 nM T77365 CKN9Y0 135543763 Ki = 25 nM T77365 C6WLJ3 135544018 IC50 > 10000 nM T77365 C1K5QE 135544028 IC50 > 10000 nM T77365 CMOB21 135544044 IC50 > 10000 nM T77365 CR6X3F 135544059 IC50 > 10000 nM T77365 C38LZC 135545353 Ki > 1000 nM T77365 CI3LK7 135546224 Ki = 210 nM T77365 C5Y9WX 135546648 Ki > 1000 nM T77365 CESD69 135546649 Ki > 1000 nM T77365 CUI90X 135546657 Ki > 1000 nM T77365 C5KX8N 135546658 Ki > 1000 nM T77365 CNCD32 135566609 Ki = 1.413 nM T77365 C8LBZ5 135624236 Ki = 201 nM T77365 C7NR5U 135645511 Ki = 3600 nM T77365 CSO0H1 135646528 Ki > 100000 nM T77365 CWIL91 135665340 IC50 > 10000 nM T77365 C7KW6I 135678052 Ki > 1000 nM T77365 CLV18T 135738630 IC50 > 10000 nM T77365 C26YKB 135738631 IC50 = 2600 nM T77365 C27QXV 135738634 IC50 > 10000 nM T77365 C1BX3M 135738635 IC50 > 10000 nM T77365 C7EI9N 135738639 IC50 > 10000 nM T77365 CHFQ46 135738640 IC50 = 760 nM T77365 CC4D8I 135738642 IC50 > 10000 nM T77365 CE6LS4 135738644 IC50 = 130 nM T77365 C6GI3C 135738646 IC50 = 310 nM T77365 C67BTG 135738649 IC50 > 120 nM T77365 C8S9QY 135738652 IC50 > 10000 nM T77365 CP17UV 135738655 IC50 = 2700 nM T77365 CVKG20 135738656 IC50 = 5300 nM T77365 CD6GS7 135738659 IC50 = 190 nM T77365 C62PTQ 135874413 Ki > 1000 nM T77365 C87ZQJ 135874414 Ki > 1000 nM T77365 C9X1UL 135874415 Ki > 1000 nM T77365 CT40VW 135874416 Ki > 1000 nM T77365 C1V9TY 135874420 Ki > 1000 nM T77365 C1T4GB 135874421 Ki > 1000 nM T77365 CFSX68 135874422 Ki > 1000 nM T77365 CNLH54 135874423 Ki > 1000 nM T77365 C2FK6J 135874424 Ki > 1000 nM T77365 C04YTD 135874425 Ki > 1000 nM T77365 CIQ04D 135874427 Ki > 1000 nM T77365 C6TO4A 135874428 Ki > 1000 nM T77365 CO0C5V 135874429 Ki > 1000 nM T77365 C9JQ2C 135874430 Ki > 1000 nM T77365 CSOV01 135874431 Ki > 1000 nM T77365 C75TGS 135874432 Ki > 1000 nM T77365 C93GBH 135874433 Ki > 1000 nM T77365 CV7US0 135874434 Ki > 1000 nM T77365 CIVD34 135949027 Ki = 41 nM T77365 C7R9LG 136002185 Ki > 1000 nM T77365 C3BV1J 136002186 Ki > 1000 nM T77365 CSBL59 136002187 Ki > 1000 nM T77365 CGS18F 136002248 Ki > 1000 nM T77365 CUK9J5 136019511 Ki > 5000 nM T77365 CBZ1I4 136025838 Ki > 5000 nM T77365 CCS5F0 136025881 Ki = 1520 nM T77365 C2VZR6 136025990 Ki > 5000 nM T77365 CA17MI 136026025 Ki > 5000 nM T77365 C9SR2V 136026026 Ki > 5000 nM T77365 C6KNF2 136026027 Ki > 5000 nM T77365 CAG7O8 136026130 Ki = 12.59 nM T77365 CO90BT 136026133 Ki > 5000 nM T77365 CM3YH2 136026181 Ki > 5000 nM T77365 C4R5TS 136029179 Ki > 5200 nM T77365 CACT14 136029180 Ki = 4700 nM T77365 CS25RJ 136029181 Ki = 4200 nM T77365 C23ZKG 136029182 Ki = 100 nM T77365 C9WF4K 136029183 Ki = 1400 nM T77365 C5Z6AJ 136029184 Ki = 10 nM T77365 CBN0G7 136029185 Ki = 20 nM T77365 CU6TS5 136029186 Ki > 5200 nM T77365 C38LUX 136036809 Ki > 1000 nM T77365 CQ49LB 136042243 Ki = 1750 nM T77365 CEHF18 136042327 Ki > 1000 nM T77365 C4U7ZM 136042328 Ki > 1000 nM T77365 CSR0Z3 136042329 Ki > 1000 nM T77365 C9C2SF 136042330 Ki > 1000 nM T77365 C75CXE 136042331 Ki > 1000 nM T77365 CS49WL 136042332 Ki > 1000 nM T77365 CQ2ZA9 136042333 Ki > 1000 nM T77365 CON2J4 136042334 Ki > 1000 nM T77365 C5VY2Z 136042335 Ki > 1000 nM T77365 CTEB06 136042336 Ki > 1000 nM T77365 CJW64L 136042337 Ki > 1000 nM T77365 C05QUF 136042338 Ki > 1000 nM T77365 C0SX1K 136042339 Ki > 1000 nM T77365 CQ37GX 136042340 Ki > 1000 nM T77365 CF3BR5 136042341 Ki > 1000 nM T77365 C75XRI 136042342 Ki > 1000 nM T77365 CS7HM2 136042343 Ki > 1000 nM T77365 C3S1WY 136042344 Ki > 1000 nM T77365 CR5H4M 136042345 Ki > 1000 nM T77365 C29YZE 136042346 Ki > 1000 nM T77365 CAP1C6 136042347 Ki > 1000 nM T77365 C5EX7D 136042348 Ki > 1000 nM T77365 C4L7GE 136042349 Ki > 1000 nM T77365 C9JM7Y 136042350 Ki > 1000 nM T77365 CO15GM 136042351 Ki > 1000 nM T77365 COEZ25 136042352 Ki > 1000 nM T77365 CGX6H7 136042353 Ki > 1000 nM T77365 C1W9XD 136042354 Ki > 1000 nM T77365 CA6TI2 136042355 Ki > 1000 nM T77365 CJ75XH 136068601 Ki > 5000 nM T77365 CL5B7U 136068602 Ki > 5000 nM T77365 CU6C4Z 136068688 Ki > 5000 nM T77365 CSJE87 136068689 Ki > 5000 nM T77365 C7SLK3 136068716 Ki > 5000 nM T77365 CZWP52 136068717 Ki = 2010 nM T77365 CDX2Q0 136068718 Ki > 5000 nM T77365 CY1RT3 136068719 Ki > 5000 nM T77365 C2XW1I 136074047 Ki = 4.074 nM T77365 CCB5S0 136079175 Ki = 12.3 nM T77365 CRP3J2 136079180 Ki = 1 nM T77365 CQ5ME1 136079181 Ki = 1.585 nM T77365 CI1PK7 136086896 Ki > 5000 nM T77365 C5HL7K 136086897 Ki > 5000 nM T77365 C6VLR1 136086898 Ki > 5000 nM T77365 CL2E0U 136086899 Ki > 5000 nM T77365 C01GMB 136086900 Ki > 5000 nM T77365 CA3X5T 136086901 Ki > 5000 nM T77365 CW49CH 136086902 Ki > 5000 nM T77365 C4F5WR 136086903 Ki > 5000 nM T77365 CS58QU 136086904 Ki > 5000 nM T77365 C4B1TU 136086905 Ki = 2130 nM T77365 CMOR91 136086906 Ki > 5000 nM T77365 C3HY9O 136086907 Ki > 5000 nM T77365 CWF2L1 136086908 Ki > 5000 nM T77365 C2X4JG 136117757 Ki = 1.9 nM T77365 CQHW89 136184487 Ki = 12.59 nM T77365 C1OU7W 136184488 Ki = 25.12 nM T77365 CW2D5Y 136184489 Ki = 19.05 nM T77365 CI2YG5 136184490 Ki = 186.21 nM T77365 CN6RY1 136184491 Ki = 93.33 nM T77365 C8OWD1 136184493 Ki = 87.1 nM T77365 CRC2O9 136184494 Ki = 32.36 nM T77365 C5EPJ2 136199393 Ki = 2832 nM T77365 CF51IY 136228031 Ki = 8780 nM T77365 C5IX2C 136236319 Ki > 30000 nM T77365 CWL69G 136414902 Ki = 2900 nM T77365 CDZ07W 137631401 Ki = 1080 nM T77365 CY61SG 137631471 Ki = 560 nM T77365 C9QS4J 137631671 Ki >= 10000 nM T77365 CE7LZ9 137632204 Ki = 2480 nM T77365 CSM29H 137632333 Ki = 4.2 nM T77365 CQ36UP 137632356 Ki > 30000 nM T77365 CH5F6G 137632488 Ki = 11900 nM T77365 C74SZH 137632691 Ki = 2.1 nM T77365 C92FIL 137632746 Ki > 30000 nM T77365 CG0F3S 137632859 Ki = 76 nM T77365 CFWO04 137632925 Ki = 3.5 nM T77365 CJ67UL 137633007 Ki = 3480 nM T77365 C2AG4Y 137633276 Ki = 238 nM T77365 C9SYC5 137633560 Ki = 1120 nM T77365 CZ2HV1 137633654 Ki = 9430 nM T77365 CZC9A2 137633810 Ki = 1038 nM T77365 C8K7EM 137634052 EC50 = 758.58 nM T77365 C9YB3R 137634085 Ki = 2.4 nM T77365 C71MVS 137634444 EC50 = 3630.78 nM T77365 CQ6C4I 137635228 Ki = 24 nM T77365 C0X6YW 137635665 Ki = 25 nM T77365 CRGN40 137635666 Ki = 309 nM T77365 CYL3X8 137636099 EC50 = 13.3 nM T77365 CC9P6O 137636304 Ki = 0.25 nM T77365 C01OZS 137636323 Ki = 4066 nM T77365 CS1EO0 137636334 Ki = 5.1 nM T77365 CU9G8K 137636427 Ki > 30000 nM T77365 C6ABK1 137636769 Ki = 1260 nM T77365 C5P9LI 137637451 Ki = 14500 nM T77365 C53RQW 137637667 Ki = 2.9 nM T77365 C6Q9JG 137637685 Ki = 353 nM T77365 CCTH80 137638080 EC50 = 6.71 nM T77365 C91WNM 137638192 Ki = 265 nM T77365 CW4S1V 137638211 Ki = 10.6 nM T77365 C5UQ4L 137638318 Ki = 1700 nM T77365 CQ8ZL2 137638623 Ki = 138 nM T77365 CSFL97 137639308 Ki = 42 nM T77365 CZ9QX0 137639459 Ki > 30000 nM T77365 CS1K4G 137639818 Ki = 854 nM T77365 C0SC7L 137640093 Ki > 30000 nM T77365 C8SUZ2 137640569 Ki = 22 nM T77365 CA8E3Q 137640739 Ki = 55 nM T77365 C45FXO 137641603 Ki = 10200 nM T77365 CG0DI3 137641858 EC50 = 645.65 nM T77365 C52XDH 137641906 Ki = 402 nM T77365 CFW9R5 137641990 EC50 = 60.2 nM T77365 CV81KH 137642036 EC50 = 16.6 nM T77365 CE4C5Y 137642150 Ki > 30000 nM T77365 CO94EX 137642153 EC50 = 14.7 nM T77365 C1Y3WC 137642555 Ki = 29 nM T77365 CB8L7K 137642940 Ki = 899 nM T77365 C7K9ZB 137642980 Ki > 30000 nM T77365 C76XKJ 137643150 Ki = 708 nM T77365 CJQD73 137643164 EC50 = 1318.26 nM T77365 CBL2G5 137643847 Ki = 58 nM T77365 CG46DW 137644190 Ki = 78 nM T77365 CPR72G 137644224 Ki = 415 nM T77365 C4R0OC 137644481 Ki > 30000 nM T77365 CY9L7W 137644817 Ki = 1 nM T77365 CI7B3F 137645065 Ki = 5090 nM T77365 CGLI82 137645223 Ki = 1960 nM T77365 CF09IY 137645275 Ki > 30000 nM T77365 C7A4FB 137645645 Ki = 51 nM T77365 CCW5R0 137645696 Ki = 1160 nM T77365 CDBT79 137645728 Ki = 10 nM T77365 C95UJV 137645798 Ki > 30000 nM T77365 CJ20CU 137645935 Ki = 3.4 nM T77365 C8YN3Q 137646655 EC50 = 2691.53 nM T77365 CER23T 137646828 EC50 = 56.23 nM T77365 CGL83H 137647102 Ki > 30000 nM T77365 CC0UF1 137647420 EC50 = 4.46 nM T77365 CT91AP 137648111 Ki = 45 nM T77365 CCA7I4 137648143 Ki = 387 nM T77365 CRK65V 137648326 Ki = 13 nM T77365 C1AIP8 137648928 EC50 = 2.87 nM T77365 CS3DT1 137649083 EC50 = 144.54 nM T77365 CWH89G 137649841 EC50 = 436.52 nM T77365 CF8W4J 137650092 Ki = 5.4 nM T77365 CIE03Y 137650221 EC50 = 38.4 nM T77365 C0XZT2 137650223 Ki = 12 nM T77365 C9W3PX 137650461 EC50 = 2344.23 nM T77365 CIM50G 137650899 EC50 = 54.3 nM T77365 CXCA79 137650918 EC50 = 354.81 nM T77365 CH8Y1E 137651023 Ki = 39.7 nM T77365 C26YKP 137651319 Ki = 7.2 nM T77365 CEAU34 137651531 Ki = 5870 nM T77365 C13AMI 137651532 Ki = 7.4 nM T77365 C6AR5M 137651599 Ki = 21 nM T77365 C9M7QE 137651747 EC50 = 31.3 nM T77365 C52VBU 137651751 Ki = 1200 nM T77365 C6Z1HJ 137651756 Ki = 10400 nM T77365 C9G7TP 137652167 Ki = 1350 nM T77365 CVS93H 137652383 Ki > 100000 nM T77365 C8T2HN 137652475 EC50 = 4897.79 nM T77365 CJ24ZP 137653290 Ki = 232 nM T77365 CHYT41 137653409 EC50 = 1071.52 nM T77365 CJ1R9K 137653588 Ki = 19600 nM T77365 C0I1HF 137654317 Ki = 0.95 nM T77365 C8ZDS9 137654513 Ki = 1.8 nM T77365 C4VJ5C 137654976 Ki = 1090 nM T77365 C3AE6C 137655247 Ki = 555 nM T77365 C08CZX 137655429 Ki = 42 nM T77365 CA24YS 137656139 Ki = 28600 nM T77365 CGZV06 137656746 Ki = 14 nM T77365 C28GAV 137656845 EC50 = 2884.03 nM T77365 CJUE21 137656913 Ki = 8680 nM T77365 C08KJH 137657382 Ki = 4320 nM T77365 CH8PL9 137657570 Ki = 6830 nM T77365 CW07LP 137657589 Ki = 195 nM T77365 C1R4SN 137657721 Ki = 1520 nM T77365 CNTX97 137657841 EC50 = 40.7 nM T77365 CJ8BC7 137657926 EC50 = 28.6 nM T77365 CQ9BR1 137658051 Ki = 485 nM T77365 C4XSN0 137658330 Ki = 310 nM T77365 C05LZQ 137658498 Ki = 2.6 nM T77365 CH9A8M 137658761 Ki = 1360 nM T77365 CRH98I 137658892 Ki = 520 nM T77365 CV7UE3 137659204 Ki = 1319 nM T77365 CY67UM 137659236 Ki > 30000 nM T77365 C2TSN7 137659296 Ki = 15 nM T77365 CO6B8M 137659407 Ki = 1230 nM T77365 C8NPD1 137659423 Ki = 4.7 nM T77365 C7VNS4 137659441 EC50 = 14.4 nM T77365 CT23EA 137659930 Ki = 6.8 nM T77365 C1NZL8 137659963 Ki > 30000 nM T77365 C3Y2IZ 137661132 EC50 = 16 nM T77365 CFUM75 137661322 Ki = 10500 nM T77365 C26LVX 137661505 EC50 = 147.91 nM T77365 C1DL4J 137661670 EC50 = 96.5 nM T77365 CBVZ04 137661692 Ki = 500 nM T77365 COM9G6 137661811 Ki > 30000 nM T77365 CD1Z9C 137661874 Ki = 1.1 nM T77365 CU1K4Z 137661957 Ki = 2.1 nM T77365 CP02WU 139030524 Ki = 68 nM T77365 CU3PW1 139248507 Ki > 1000 nM T77365 CT1H6B 139248508 Ki > 1000 nM T77365 CUIN96 139248509 Ki > 1000 nM T77365 CW74BD 141536950 Ki = 55300 nM T77365 C6SUZ3 143294251 Ki = 307 nM T77365 CN2LX1 144852560 Ki = 1340 nM T77365 CBV2L5 145436760 IC50 = 0.0017 nM T77365 CK15TH 145436761 Ki = 5.14 nM T77365 C6KOB8 145436762 Ki = 2.15 nM T77365 CM7J2Q 145436763 Ki = 0.24 nM T77365 CSQL37 145436764 Ki = 0.25 nM T77365 CNP52A 145436765 IC50 = 0.045 nM T77365 C6OFP7 145436766 Ki = 0.42 nM T77365 CSQ8U5 145436767 IC50 = 0.011 nM T77365 C4PZ5S 145436769 IC50 = 0.0016 nM T77365 CORZ59 145948563 IC50 = 1071.52 nM T77365 CI75YJ 145949481 Ki = 34 nM T77365 CZ0XE2 145951783 Ki = 0.6166 nM T77365 CJM3T1 145952643 Ki > 10000 nM T77365 CUO32M 145953622 Ki = 1.514 nM T77365 C2GVM4 145954098 Ki = 10.1 nM T77365 C8VS3W 145954236 Ki > 10000 nM T77365 CQ9G0K 145954398 Ki = 20 nM T77365 C3RU6S 145954471 Ki = 144 nM T77365 CZX79R 145954995 Ki > 100000 nM T77365 C6V4WO 145957791 Ki = 0.8913 nM T77365 CC0OX1 145958464 Ki = 2.24 nM T77365 CI7EA2 145958874 Ki = 1.023 nM T77365 CH7G6S 145960536 Ki = 532 nM T77365 CW45RB 145960619 Ki = 3141 nM T77365 C9PT5Q 145960667 Ki = 78 nM T77365 C3BY8E 145960746 Ki = 973 nM T77365 C9ZND4 145960774 Ki = 238 nM T77365 CWSM81 145960813 Ki = 28 nM T77365 C5D6AI 145960873 Ki = 406 nM T77365 C62JCL 145960933 Ki = 99 nM T77365 C59ASP 145961050 Ki = 23 nM T77365 CQN69Z 145961145 Ki = 2487 nM T77365 CRBY29 145961339 Ki = 608 nM T77365 CJE0K4 145961433 Ki > 10000 nM T77365 CTV13K 145961745 Ki > 10000 nM T77365 C2BZ5C 145961747 Ki = 630 nM T77365 C02OQR 145961748 Ki = 79 nM T77365 C1O0GQ 145961937 Ki = 219 nM T77365 CTRZ67 145961995 Ki = 530 nM T77365 CCB0Y2 145961997 Ki = 212 nM T77365 CT8UO0 145962202 Ki = 42 nM T77365 C3M7ZN 145962234 Ki = 403 nM T77365 C9DHW0 145962261 Ki = 117 nM T77365 CL79QC 145962272 Ki = 1630 nM T77365 CVA89T 145962310 Ki = 96 nM T77365 C4YHU8 145962337 Ki > 10000 nM T77365 CD6X5O 145962355 Ki = 4.72 nM T77365 C86APL 145962364 Ki = 313 nM T77365 CH5DS7 145962529 Ki = 61 nM T77365 CN0RW5 145962558 Ki > 10000 nM T77365 CJH4A7 145962653 Ki = 2869 nM T77365 C4NXC1 145962657 Ki > 10000 nM T77365 CN0AG6 145962770 Ki = 3392 nM T77365 CH6J9M 145962802 Ki > 10000 nM T77365 CLB9Q2 145962957 Ki = 250 nM T77365 C8MFE6 145963003 Ki > 10000 nM T77365 C9LHF2 145963054 Ki > 10000 nM T77365 CG6U5V 145963081 Ki > 10000 nM T77365 C9UYI6 145963230 Ki = 116 nM T77365 CYK7D8 145963377 Ki > 10000 nM T77365 CLBR08 145963459 Ki = 418 nM T77365 CU12MA 145963481 Ki = 2000 nM T77365 C2WR5P 145963553 Ki > 10000 nM T77365 C5MD4S 145963661 Ki = 135 nM T77365 CZ98EW 145963678 Ki > 10000 nM T77365 CVH6D7 145964038 Ki = 0.4 nM T77365 C01PVB 145965471 Ki = 221 nM T77365 C1ER6I 145967791 Ki = 58.7 nM T77365 C8J7FL 145971923 Ki = 12 nM T77365 CZJA45 145972655 Ki = 22 nM T77365 CE23KG 145973077 Ki = 764 nM T77365 CV9OM2 145973260 Ki = 0.4 nM T77365 CBT7E9 145973326 Ki = 1600 nM T77365 CI2HN1 145977111 Ki > 10000 nM T77365 C8W0MQ 145978569 Ki = 424 nM T77365 C3M7CX 145978972 Ki = 332 nM T77365 C17MYD 145979308 Ki = 81 nM T77365 C3JE4Q 145979392 Ki > 10000 nM T77365 CI26CB 145979547 Ki = 438 nM T77365 C5SZN2 145979632 Ki = 827 nM T77365 C43NUZ 145980000 Ki = 6.36 nM T77365 C0GMD9 145980280 Ki > 10000 nM T77365 COK2V5 145980546 Ki = 47.6 nM T77365 CO3Y8B 145980553 Ki = 12400 nM T77365 CP92RY 145980571 Ki = 7410 nM T77365 C7NJH2 145980712 Ki = 194 nM T77365 CMFW02 145980971 Ki = 15.7 nM T77365 CDM63O 145981315 Ki = 37.2 nM T77365 CHQ73C 145981492 Ki = 342 nM T77365 CA9R1X 145981583 Ki = 18.6 nM T77365 CC1I0V 145981690 Ki = 1000 nM T77365 CX02DQ 145981864 Ki = 62.2 nM T77365 CNTY13 145982075 Ki = 14.9 nM T77365 CAI53J 145982270 Ki = 24.3 nM T77365 CI35AM 145982396 Ki = 202 nM T77365 CHSJ14 145982423 Ki = 829 nM T77365 C8RT4W 145982945 Ki = 169 nM T77365 C0QSZ6 145983668 Ki = 90 nM T77365 C9CG6I 145984161 Ki = 34000 nM T77365 CUM74P 145984609 Ki = 1540 nM T77365 C9VDN3 145985635 Ki = 10300 nM T77365 C19BNU 145986670 Ki = 8040 nM T77365 CQ9AK0 145987082 Ki = 197 nM T77365 C15LTN 145987104 Ki = 98 nM T77365 CJ70FS 145987226 Ki = 86.5 nM T77365 C3A0XB 145987543 Ki = 295 nM T77365 C05IZF 145987813 Ki > 100000 nM T77365 CGV37C 145987819 Ki = 11 nM T77365 CFNH51 145987858 Ki > 10000 nM T77365 CT79VE 145988064 Ki = 135 nM T77365 C0AF1D 145988094 Ki = 32.5 nM T77365 C2NB1M 145988388 Ki = 30 nM T77365 CD01TO 145988590 Ki = 22.8 nM T77365 C3O1MT 145988709 Ki = 6.24 nM T77365 CMD74V 145988733 Ki = 38.2 nM T77365 CV53QZ 145988884 Ki = 9.29 nM T77365 C8CO2G 145989004 Ki > 10000 nM T77365 CEM2L0 145989440 Ki = 137 nM T77365 CVS17Y 145989611 Ki = 2950 nM T77365 C8IZN5 145989729 Ki > 10000 nM T77365 CB9GL1 145989764 Ki = 16700 nM T77365 C4I1EY 145990207 Ki = 9390 nM T77365 C98GKM 145990252 Ki = 30.3 nM T77365 C5E2PC 145990255 Ki = 210 nM T77365 CZP5T3 145990301 Ki = 1860 nM T77365 CJ0A5L 145990511 Ki = 13000 nM T77365 CHV8C9 145990554 Ki = 6.12 nM T77365 C3H2ZP 145990725 Ki = 32 nM T77365 CJ30YT 145990769 Ki = 81.3 nM T77365 CC4BW2 145990800 Ki = 40 nM T77365 C2Y8PA 145990926 Ki = 11200 nM T77365 CV5XO6 145991048 Ki = 141 nM T77365 C6ZYL7 145991283 Ki = 41.8 nM T77365 C9YO2T 145991303 Ki = 63.1 nM T77365 CRJ65G 145991313 Ki = 90 nM T77365 CN7A1X 145991427 Ki = 13400 nM T77365 CUYV92 145991447 IC50 = 250 nM T77365 CUP48Y 145991545 Ki = 21 nM T77365 C8QT3X 145991607 Ki = 11800 nM T77365 C7K5ZQ 145991651 Ki = 22600 nM T77365 C8SI9A 145991749 Ki = 114 nM T77365 C2CB3J 145991827 Ki = 59.4 nM T77365 CFH29P 145992091 Ki > 10000 nM T77365 C3QHT6 145992189 Ki = 71.9 nM T77365 C1MU4D 145992652 Ki = 100 nM T77365 CB85AS 145992677 Ki = 8840 nM T77365 C94OJE 145992790 Ki = 71.5 nM T77365 C7B3FY 145992928 Ki = 29.7 nM T77365 C47DOA 145993092 Ki > 30000 nM T77365 CZOR31 145993511 Ki = 13.2 nM T77365 CQ93KE 145993540 Ki = 6.46 nM T77365 CW36TA 145993667 Ki = 24.6 nM T77365 CC2I1H 145993863 Ki = 71 nM T77365 C6A3RN 145993941 Ki = 21 nM T77365 CO69HC 145994068 Ki > 100000 nM T77365 C72SMW 145994175 Ki = 376 nM T77365 CE07TR 145994259 Ki = 61.6 nM T77365 C5LXC4 153605593 Ki = 3550 nM T77365 CZ53NG 153605599 Ki = 2550 nM T77365 C4W8PK 155413621 Ki = 216 nM T77365 C2CG8J 155510487 Ki = 3240 nM T77365 C14XVK 155510489 Ki = 3.4 nM T77365 CEXH54 155511332 EC50 = 10.15 nM T77365 CD52TC 155511687 Ki = 1951 nM T77365 C0TVO4 155511832 Ki = 300 nM T77365 CPMN94 155511844 Ki = 114 nM T77365 C4FA0V 155512157 Ki = 1306 nM T77365 CM5ZA9 155512438 Ki = 131 nM T77365 CX96QM 155512576 Ki = 21400 nM T77365 CLUF91 155513199 EC50 = 1.38 nM T77365 CV35ZN 155513505 Ki = 5200 nM T77365 CGS27D 155513515 Ki = 2.36 nM T77365 CV20JC 155513938 Ki = 6625 nM T77365 CP7UX3 155513958 Ki = 1258.93 nM T77365 CUB2C9 155514153 Ki = 887 nM T77365 C38LUS 155514209 Ki = 26 nM T77365 CST9B5 155514281 Ki = 6276 nM T77365 CR85FY 155514357 Ki = 195 nM T77365 CQ7GR6 155514463 Ki = 1.7 nM T77365 CF04MH 155514522 Ki = 800 nM T77365 CGIT15 155514690 Ki > 10000 nM T77365 CRF2B1 155514696 Ki = 24 nM T77365 CN8E1J 155514860 Ki = 189 nM T77365 CP6C5S 155514957 Ki = 204 nM T77365 CLJ7Y3 155515226 Ki = 682 nM T77365 CNV02U 155516016 Ki = 8860 nM T77365 CT18NO 155516071 Ki = 0.59 nM T77365 CLX4D7 155516277 Ki = 140 nM T77365 CR59VH 155517789 Ki = 53 nM T77365 C0CR9Q 155518147 Ki = 168 nM T77365 C2PM8H 155518462 Ki > 10000 nM T77365 CR40UE 155518944 EC50 = 1.1 nM T77365 CP74IJ 155519148 Ki = 2.4 nM T77365 CX1MO3 155519551 Ki = 108 nM T77365 C5YDE2 155519621 Ki = 2370 nM T77365 CEY82J 155519727 Ki > 30000 nM T77365 C5NTJ8 155519776 Ki = 5 nM T77365 C72OJY 155519986 Ki = 2.4 nM T77365 C8N1CQ 155520115 Ki = 5 nM T77365 CXS1T4 155520635 Ki = 801 nM T77365 CZ1S5N 155520662 Ki = 22.4 nM T77365 CPL4Q7 155520955 Ki = 94.5 nM T77365 C6A4UH 155521103 Ki = 33.6 nM T77365 CS2GJ8 155521355 Ki = 3980 nM T77365 C25KBM 155521478 Ki > 30000 nM T77365 C1LH7J 155521488 Ki = 239 nM T77365 CYW7Q0 155521543 Ki = 89.5 nM T77365 CW29KY 155521694 Ki = 1.8 nM T77365 CHTX98 155522541 Ki = 245 nM T77365 CSBN54 155522680 Ki = 208 nM T77365 CGJ0W4 155522875 Ki = 36.4 nM T77365 CBW5G4 155522899 Ki = 11.2 nM T77365 C3SJ9B 155523748 Ki = 248 nM T77365 CK8RS0 155523968 Ki = 40.7 nM T77365 C4ZIH2 155524032 Ki = 2990 nM T77365 CMLS87 155524113 EC50 = 4.6 nM T77365 C8E3HR 155524516 Ki = 140 nM T77365 CYSK39 155525038 Ki = 1144 nM T77365 CZX2N4 155525050 Ki = 197 nM T77365 CN1C6R 155525265 Ki = 16.8 nM T77365 C8QIF6 155525396 Ki = 100 nM T77365 C78DHT 155525494 Ki = 0.17 nM T77365 CR6A7N 155525747 Ki = 1.9 nM T77365 CT24MQ 155526752 EC50 = 5.52 nM T77365 CBAK91 155527112 Ki = 169 nM T77365 CS9U0T 155527740 Ki = 2.5 nM T77365 C15MXV 155527829 Ki = 61 nM T77365 C3KA0S 155528136 Ki = 1000 nM T77365 CHR60D 155528366 IC50 = 910 nM T77365 CAR75Z 155528717 Ki > 1000 nM T77365 CZ53GQ 155528757 Ki = 624 nM T77365 CXM9W5 155529088 Ki = 6309.57 nM T77365 CZWH28 155529694 Ki = 173 nM T77365 CZ9YC8 155529872 Ki = 35.3 nM T77365 CVE30Z 155530257 Ki = 135 nM T77365 CS2BT0 155530292 Ki = 520 nM T77365 CQT8O2 155530381 Ki > 1000 nM T77365 C78JZY 155530514 Ki = 92.4 nM T77365 C4L7ZO 155530653 IC50 = 520 nM T77365 CN87UW 155530961 Ki = 800 nM T77365 CNVU03 155531548 Ki = 109.8 nM T77365 C3XQ9S 155531570 Ki = 14.9 nM T77365 C4A3DX 155531727 Ki > 1000 nM T77365 C14GCE 155531842 Ki = 5850 nM T77365 CQI01K 155531990 Ki > 1000 nM T77365 C7A9BH 155532173 Ki = 3 nM T77365 C21MLU 155532274 Ki > 1000 nM T77365 CVI21H 155532514 Ki = 160 nM T77365 C86SCT 155532773 Ki = 14750 nM T77365 CJH8R0 155532913 Ki = 71 nM T77365 CQ96YB 155532918 Ki = 2170 nM T77365 C9EU2D 155533104 Ki > 100000 nM T77365 CY8O6B 155533349 Ki = 52.6 nM T77365 C03YFW 155533388 Ki = 8.3 nM T77365 C7E5OP 155533880 Ki = 314 nM T77365 CH54UR 155534188 Ki = 674 nM T77365 CW8FN0 155534473 Ki = 104 nM T77365 C9QV4W 155534659 Ki = 7.7 nM T77365 C4NU8B 155534836 Ki = 108 nM T77365 C9ZK5A 155535230 EC50 = 0.64 nM T77365 C67VZK 155535458 Ki = 16100 nM T77365 CH6E1O 155536745 Ki = 357 nM T77365 C6Q1EM 155536934 Ki = 756 nM T77365 C3P8VK 155537874 Ki = 6010 nM T77365 CSMI71 155540479 IC50 = 420 nM T77365 C8BHN2 155540525 Ki = 3.5 nM T77365 CF6ZE5 155540615 Ki = 363 nM T77365 C3P1ZT 155540839 Ki = 1580 nM T77365 C2L9TS 155540948 Ki > 1000 nM T77365 C4KDO9 155541051 Ki = 693 nM T77365 C19HQM 155541262 Ki = 8910 nM T77365 C2HX6J 155541790 Ki = 7.4 nM T77365 C9H5VC 155541975 Ki > 100000 nM T77365 CQ1FY8 155542311 Ki = 636 nM T77365 CMEW36 155542520 Ki = 93 nM T77365 CGY1J4 155542588 Ki = 233 nM T77365 CCV87Q 155542600 Ki > 1000 nM T77365 C8JY0G 155542643 Ki = 189 nM T77365 C0BFX9 155542720 Ki = 1160 nM T77365 C06OKY 155542884 Ki = 82 nM T77365 CR8A7D 155543424 Ki = 101 nM T77365 C3XDT7 155543719 Ki = 19 nM T77365 C2DNQ0 155543871 Ki = 32900 nM T77365 C1QAZ9 155544096 Ki = 346 nM T77365 CR0EV6 155544177 Ki > 100000 nM T77365 C30NOS 155544777 Ki = 3040 nM T77365 CQ9Z2P 155545386 Ki = 1.64 nM T77365 C5Y4BH 155545414 Ki = 1510 nM T77365 C5HU6A 155545585 Ki = 241 nM T77365 C45CUJ 155545762 Ki > 1000 nM T77365 CM5ZN0 155545870 Ki = 650 nM T77365 C2NKO5 155545904 Ki = 428 nM T77365 C3B0SI 155546100 Ki = 2.1 nM T77365 C95ICF 155546118 Ki = 3900 nM T77365 C4BHE8 155546183 Ki = 1080000 nM T77365 CL1T9K 155546550 Ki = 5.2 nM T77365 C6XP3U 155546562 Ki > 1000 nM T77365 CHC2O5 155547064 Ki = 8.5 nM T77365 C1VHM5 155547186 Ki = 64400 nM T77365 CQE30Y 155547305 Ki = 1260 nM T77365 CK1X5S 155547588 Ki = 8270 nM T77365 C8Q7JG 155547782 Ki = 1610 nM T77365 C35WAK 155548264 Ki > 1000 nM T77365 C39GTQ 155548778 Ki = 115.3 nM T77365 CY1XJ0 155548779 Ki > 100000 nM T77365 C4MIT2 155548780 Ki = 1700 nM T77365 C82STM 155549033 Ki = 3162.28 nM T77365 C3NE6F 155549264 Ki = 93.8 nM T77365 CY5U1J 155549967 Ki = 224 nM T77365 CC45SE 155550088 Ki = 1210 nM T77365 CY7Q9N 155550159 Ki = 77.8 nM T77365 C2IU1J 155550532 Ki = 959 nM T77365 C6J5EX 155550807 Ki = 217 nM T77365 CN2I3H 155550832 Ki = 12900 nM T77365 CT7MV5 155551482 Ki = 1329 nM T77365 C41JXM 155551530 Ki = 67 nM T77365 C4LN3W 155551750 Ki = 314 nM T77365 CI41QF 155552117 Ki = 1750 nM T77365 CA29GP 155552390 Ki = 7.7 nM T77365 CJ82KN 155552405 Ki = 143 nM T77365 CM40UT 155552539 Ki > 1000 nM T77365 CIQH30 155552719 Ki > 1000 nM T77365 CX4P7S 155553385 Ki > 100000 nM T77365 CD42WK 155553510 Ki = 5.7 nM T77365 CNK6Z9 155553575 Ki = 322 nM T77365 CY08CH 155553600 Ki = 1622 nM T77365 CB75AP 155553750 Ki > 1000 nM T77365 CG1CF2 155553962 EC50 = 4.05 nM T77365 CU1ZE5 155554091 IC50 = 58 nM T77365 CFW01A 155554317 Ki > 30000 nM T77365 CPXQ16 155554464 IC50 = 22 nM T77365 C57MKC 155555241 Ki = 881 nM T77365 CWCN91 155555408 Ki = 1449 nM T77365 CVDO87 155555721 Ki > 1000 nM T77365 CN38KO 155555854 Ki = 21100 nM T77365 CL3IB5 155555868 Ki = 348 nM T77365 CJ73SL 155556032 Ki = 784 nM T77365 CDR63F 155556134 Ki > 30000 nM T77365 CYB6T5 155556258 Ki = 4060 nM T77365 CV9P2M 155556457 Ki = 346 nM T77365 CC14ON 155556524 Ki > 1000 nM T77365 C7M1VE 155556836 Ki = 25900 nM T77365 CGF0H2 155556884 Ki > 1000 nM T77365 C2F1JY 155557284 Ki = 5690 nM T77365 CTSX95 155557611 Ki = 1020 nM T77365 CJ16GB 155557960 Ki = 767 nM T77365 C7FUQ6 155558172 Ki = 461 nM T77365 C0W7AL 155558312 Ki = 512 nM T77365 CDMC47 155558350 Ki = 141.6 nM T77365 C3A7MK 155558447 Ki > 1000 nM T77365 C8Z2TC 155558489 Ki = 1060 nM T77365 CYX8T1 155558921 Ki = 1340 nM T77365 CIAE48 155558941 Ki = 8.5 nM T77365 CVS4T6 155559056 Ki > 100000 nM T77365 CDZX46 155559070 Ki = 96 nM T77365 CTI57G 155559203 Ki > 1000 nM T77365 CP87XK 155559423 Ki = 369 nM T77365 CMU6P5 155559511 Ki = 1330 nM T77365 CQM64H 155559636 Ki = 22.9 nM T77365 CV5PC7 155559963 EC50 = 5.7 nM T77365 C34ORN 155560261 Ki > 100000 nM T77365 C8B7CG 155560391 Ki > 1000 nM T77365 C73XYW 155560510 Ki = 208 nM T77365 C3OP1F 155560545 Ki > 1000 nM T77365 CEXP80 155561009 Ki > 1000 nM T77365 C5KY7D 155561141 Ki = 403 nM T77365 CGD7R4 155561189 Ki = 52.7 nM T77365 CQ2L0P 155561909 Ki = 6.4 nM T77365 CKG56Z 155562044 Ki = 313 nM T77365 CXUN73 155562096 Ki = 581 nM T77365 C6EN2B 155562182 Ki = 96.7 nM T77365 C5X9FM 155562751 Ki = 5495 nM T77365 C1NF2M 155562789 Ki = 627 nM T77365 CM46KC 155563177 Ki > 1000 nM T77365 CQ19VC 155563189 Ki = 887 nM T77365 CJZO26 155563438 Ki > 100000 nM T77365 CPTM25 155563673 Ki = 8000 nM T77365 C5ZKN0 155563788 Ki = 2020 nM T77365 CE2V5Y 155564179 Ki > 1000 nM T77365 C8TL6J 155564465 Ki = 122 nM T77365 CHJ5Q8 155564753 Ki = 8.2 nM T77365 CFNC10 155565326 Ki = 5400 nM T77365 C8N3PQ 155565636 Ki > 1000 nM T77365 CYI54E 155565672 Ki > 1000 nM T77365 CI2CQ0 155565683 Ki > 1000 nM T77365 CB14WJ 155565911 Ki >= 1000 nM T77365 C6DQ1K 155566338 Ki = 4260 nM T77365 C0VUO9 155566764 Ki = 293 nM T77365 CN8RL3 155567003 Ki = 54.5 nM T77365 CPW8M5 155567457 Ki = 7070 nM T77365 C5KNM6 155569051 Ki = 253 nM T77365 CH86AJ 155569073 Ki > 1000 nM T77365 CP9TR0 10324985 Ki > 10000 nM T77365 C7Q9WY 11395785 Ki = 2050 nM T77365 CP2EI0 118725998 IC50 = 18 nM T77365 CFS9W4 118726022 IC50 = 1479 nM T77365 C4EBT3 16109359 EC50 = 173.78 nM T77365 CJZ23T 44333154 Ki = 6083 nM T77365 CIU68M 44333155 Ki > 10000 nM T77365 CV8BQ7 44333404 Ki = 6750 nM T77365 C30UYD 44333842 Ki = 5096 nM T77365 CCK07J 44333843 Ki = 6100 nM T77365 C90IQB 46905977 Ki = 1760 nM T77365 D00ASZ 16204411 Ki = 95 nM T77365 D00CJJ 12016636 Ki = 4900 nM T77365 D00GNW 16109429 Ki = 247 nM T77365 D00GQI 11313151 Ki = 376 nM T77365 D00HYS 18507264 Ki = 22.7 nM T77365 D00JBC 12905389 EC50 = 7600 nM T77365 D00JMT 210332 Ki > 10000 nM T77365 D00JWA 46880333 Ki = 209 nM T77365 D00MFV 44572293 Ki = 16000 nM T77365 D00MPA 9834240 Ki = 261 nM T77365 D00NFW 16109432 Ki = 177 nM T77365 D00NYG 2303947 Ki = 19 nM T77365 D00OFN 44420099 Ki = 5 nM T77365 D00TQR 86344 EC50 = 1600 nM T77365 D00YOM 15557795 Ki = 3330 nM T77365 D00YXE 11652061 Ki > 10000 nM T77365 D01CQU 5139184 Ki = 112 nM T77365 D01MOQ 13155595 Ki = 900 nM T77365 D01NHH 16109434 Ki = 1055 nM T77365 D01PGY 10045125 Ki = 267 nM T77365 D01QBK 44572356 Ki = 15000 nM T77365 D01QYQ 6603931 Ki > 260 nM T77365 D01VEU 44300688 Ki = 600 nM T77365 D01VJT 3890693 Ki = 1900 nM T77365 D01VXC 11278089 Ki = 554 nM T77365 D01VXP 16115754 Ki = 3140 nM T77365 D01WNA 5248753 Ki = 52 nM T77365 D02BGA 9877796 Ki = 46.3 nM T77365 D02EAO 11243768 Ki = 1700 nM T77365 D02FLH 16109427 Ki = 114 nM T77365 D02HOL 11849871 Ki = 300 nM T77365 D02HYT 11438116 Ki = 81.9 nM T77365 D02JCM 9841284 Ki = 750 nM T77365 D02JMR 16202727 Ki = 29.3 nM T77365 D02NBB 44449695 Ki = 85 nM T77365 D02RBK 9904551 Ki = 6100 nM T77365 D02TEW 10754789 Ki = 329 nM T77365 D02UHS 10391971 Ki = 18.9 nM T77365 D02XMQ 8321 Ki = 530 nM T77365 D02XPR 73124 Ki = 8500 nM T77365 D02YIW 1794 IC50 = 5100 nM T77365 D02ZZQ 44567454 Ki = 44100 nM T77365 D03FVK 16115753 Ki = 6310 nM T77365 D03HBG 16203543 Ki = 39.7 nM T77365 D03JFX 7 Ki = 2200 nM T77365 D03KKK 169317 EC50 = 50 nM T77365 D03LJX 651586 Ki = 2200 nM T77365 D03NVE 10226014 Ki > 5000 nM T77365 D03POP 44420681 Ki = 4290 nM T77365 D03RFA 657378 Ki = 385 nM T77365 D04AGC 18511481 Ki = 9524 nM T77365 D04DVT 126079 Ki = 595 nM T77365 D04JDQ 44401799 Ki = 270.5 nM T77365 D04JIR 69689 Ki = 6900 nM T77365 D04LZN 44572409 Ki = 660 nM T77365 D04MMG 25104891 Ki = 1900 nM T77365 D04PJO 10612371 Ki = 228 nM T77365 D04TTP 127993 Ki = 4920 nM T77365 D04WBU 12905388 EC50 = 15200 nM T77365 D04WHE 247436 Ki = 9600 nM T77365 D04XLX 44449523 Ki = 17 nM T77365 D04YUM 75929 Ki = 7800 nM T77365 D04ZTH 2817024 Ki = 32 nM T77365 D05KEF 44418996 Ki = 189 nM T77365 D05MCK 6105572 Ki = 100 nM T77365 D05OUG 2833773 Ki = 1000 nM T77365 D05SYY 10402581 Ki = 66 nM T77365 D05TFM 44449741 Ki = 30 nM T77365 D05XGF 44186581 Ki = 333 nM T77365 D05ZRR 9836155 Ki = 23 nM T77365 D05ZUX 44207909 Ki >= 1000 nM T77365 D06GOE 135465785 Ki > 1000 nM T77365 D06GTI 135416058 Ki > 1000 nM T77365 D06KYP 44572292 Ki = 74 nM T77365 D06NQD 695136 Ki = 118 nM T77365 D06PYV 11976150 Ki = 800 nM T77365 D06QRI 10378184 Ki = 1300 nM T77365 D06RCT 16203429 Ki = 45 nM T77365 D06SGU 11774068 Ki > 5000 nM T77365 D06ZWQ 4962866 Ki = 8600 nM T77365 D07DOE 44447542 Ki > 100000 nM T77365 D07FZA 135522368 Ki > 1000 nM T77365 D07HVJ 16203666 Ki = 3870 nM T77365 D07IPZ 11740439 Ki = 758 nM T77365 D07YKU 44449258 Ki = 69 nM T77365 D08AJS 135407706 Ki > 10000 nM T77365 D08AXT 44449696 Ki = 372 nM T77365 D08CIY 11424684 Ki = 2.9 nM T77365 D08EBT 10981286 Ki = 1230 nM T77365 D08EZI 11739042 Ki = 157 nM T77365 D08FOT 5311479 Ki = 3790 nM T77365 D08HBH 11359018 Ki = 103 nM T77365 D08INY 619020 Ki = 169 nM T77365 D08JUQ 11652153 Ki = 289 nM T77365 D08JYX 11743895 Ki = 2680 nM T77365 D08LZN 11450197 Ki = 14000 nM T77365 D08RGW 44403594 Ki = 9140 nM T77365 D08SJF 44403591 Ki = 3360 nM T77365 D09HAM 10491577 Ki = 91 nM T77365 D09IRV 11523232 Ki = 118 nM T77365 D09KUY 12431921 Ki > 10000 nM T77365 D09RKX 135433658 Ki > 1280 nM T77365 D09UDF 44449257 Ki = 391 nM T77365 D09VOP 16203665 Ki = 1400 nM T77365 D09VRX 11521761 Ki = 833 nM T77365 D0A0VT 44572291 Ki = 18000 nM T77365 D0A2WH 14969715 EC50 = 43400 nM T77365 D0A4MK 135489238 Ki > 1000 nM T77365 D0A6IO 5310960 Ki = 140 nM T77365 D0A6JX 452612 Ki = 4800 nM T77365 D0A9BZ 11605883 Ki = 484 nM T77365 D0AI8F 12016633 Ki = 1900 nM T77365 D0B0QW 10389852 Ki = 6520 nM T77365 D0B0TX 44572355 Ki = 6000 nM T77365 D0B2NE 44598833 Ki = 41700 nM T77365 D0B3UE 12852 Ki = 1800 nM T77365 D0B8RQ 11427528 Ki = 899 nM T77365 D0BC7P 3355253 Ki = 54 nM T77365 D0C1PS 12486289 Ki = 3900 nM T77365 D0C2UJ 8974 Ki = 120 nM T77365 D0C8ON 6710 Ki = 3200 nM T77365 D0CB9B 9813424 Ki = 35 nM T77365 D0CX7N 44572471 Ki = 85 nM T77365 D0D3WR 44401938 Ki = 34.9 nM T77365 D0D4NS 11536096 Ki > 10000 nM T77365 D0DB7A 414707 Ki = 4100 nM T77365 D0E2FV 309375 Ki = 9600 nM T77365 D0E4LB 16115752 Ki = 1820 nM T77365 D0E4UT 13789211 Ki = 8500 nM T77365 D0E5QE 25113696 Ki = 24900 nM T77365 D0E7YE 11462181 Ki = 66 nM T77365 D0E8RA 2773172 Ki = 4000 nM T77365 D0E9QX 5312112 Ki = 1800 nM T77365 D0F1AS 80220 EC50 = 75900 nM T77365 D0F4EN 11470612 Ki > 1000 nM T77365 D0F4XB 2817165 Ki = 1 nM T77365 D0FF6S 16038374 IC50 = 10000 nM T77365 D0G5ZF 10318664 Ki = 2960 nM T77365 D0G6BI 16203542 EC50 = 39.7 nM T77365 D0G6VT 16202726 Ki = 900 nM T77365 D0H5HP 17884 Ki = 250 nM T77365 D0H9BP 5697 Ki = 1 nM T77365 D0H9EY 10475082 Ki = 3.9 nM T77365 D0HK5B 9798914 Ki = 1.2 nM T77365 D0I1IW 16203539 Ki = 370 nM T77365 D0I2EQ 16109426 Ki = 375 nM T77365 D0I6MT 25104892 Ki = 4170 nM T77365 D0I7HL 14842885 Ki = 500 nM T77365 D0IG5E 44582613 Ki = 2160 nM T77365 D0J4EZ 135443359 Ki > 1000 nM T77365 D0J6ME 9964781 Ki = 13 nM T77365 D0J6PQ 44401937 Ki = 68.5 nM T77365 D0JJ6T 10021483 Ki = 1270 nM T77365 D0K0OT 1329 Ki = 56 nM T77365 D0K5WC 44567438 Ki > 100000 nM T77365 D0K6ZA 5311041 Ki = 328 nM T77365 D0K8ZZ 448222 Ki = 1 nM T77365 D0KJ3H 16203431 Ki = 373 nM T77365 D0KM0Y 10423637 Ki = 88 nM T77365 D0KT3L 10454501 Ki = 3960 nM T77365 D0L0VU 135484064 Ki > 1000 nM T77365 D0L2MN 11529627 Ki = 315 nM T77365 D0L4WN 31420 Ki = 320 nM T77365 D0L6YI 16203540 Ki = 502 nM T77365 D0LD0X 128525 EC50 = 62000 nM T77365 D0LP5V 11536936 Ki = 148 nM T77365 D0M3CG 93205 Ki = 750 nM T77365 D0N1PT 11500124 Ki > 10000 nM T77365 D0N1QO 10320311 Ki = 1780 nM T77365 D0N1QP 16109423 Ki = 39 nM T77365 D0N2DP 11484484 Ki = 46000 nM T77365 D0N2VO 668105 Ki = 130 nM T77365 D0N8RM 242652 Ki = 11000 nM T77365 D0NF3E 11565524 Ki > 10000 nM T77365 D0O0FP 9860294 Ki = 6.6 nM T77365 D0O4KI 9834769 Ki = 1.6 nM T77365 D0O6NS 81457 Ki = 3200 nM T77365 D0OR5V 414708 Ki = 2300 nM T77365 D0OX0V 11688103 Ki = 3440 nM T77365 D0P0BV 16202841 Ki = 450 nM T77365 D0P5ZE 11771279 Ki > 10000 nM T77365 D0P7FK 743242 Ki = 19 nM T77365 D0P8MK 44572469 Ki = 620 nM T77365 D0PU1R 12431922 Ki > 10000 nM T77365 D0PU6F 11658819 Ki = 561 nM T77365 D0Q1RD 16202725 Ki = 390 nM T77365 D0Q3LM 16115477 Ki = 5740 nM T77365 D0Q5HW 9801709 Ki = 35100 nM T77365 D0Q6KO 1942 Ki = 3100 nM T77365 D0Q6WX 2690 Ki = 0.142 nM T77365 D0Q9GL 135443367 Ki > 1000 nM T77365 D0QD3O 619024 Ki = 405 nM T77365 D0QN4U 16202728 Ki = 252 nM T77365 D0QN5I 9964493 Ki = 14 nM T77365 D0R1XY 123807 Ki = 17 nM T77365 D0R8OK 822296 Ki = 120 nM T77365 D0RZ2M 11572592 Ki = 53 nM T77365 D0S4JI 20262 Ki = 8500 nM T77365 D0S5XP 44572408 Ki = 730 nM T77365 D0S6QA 11608719 Ki = 730 nM T77365 D0T2RY 9948320 Ki >= 1000 nM T77365 D0TC7N 9953255 Ki = 620 nM T77365 D0TU7I 5353365 Ki = 36 nM T77365 D0UM6O 44449565 Ki = 20 nM T77365 D0UZ4J 6604926 Ki = 670 nM T77365 D0V7MX 247678 Ki = 11000 nM T77365 D0V8MD 1922 IC50 = 454 nM T77365 D0V9EE 24950370 Ki = 11 nM T77365 D0W1PF 16109428 Ki = 230 nM T77365 D0W3MT 11565892 Ki = 167 nM T77365 D0W5CZ 21976428 Ki = 242 nM T77365 D0W6FC 44572473 Ki = 1100 nM T77365 D0W6TG 44186666 Ki = 22.7 nM T77365 D0W8RB 44572357 Ki = 1600 nM T77365 D0WI4D 11617054 Ki = 55 nM T77365 D0X5PJ 135529391 Ki > 1000 nM T77365 D0Y5TL 5372720 Ki = 935 nM T77365 D0Y5WQ 44185871 Ki > 10000 nM T77365 D0Y6HQ 16115478 Ki = 12500 nM T77365 D0Y7AV 44449709 Ki = 681 nM T77365 D0Y7HG 5281616 Ki = 16700 nM T77365 D0Y8EU 393595 Ki = 25 nM T77365 D0Y8LD 135529386 Ki > 1000 nM T77365 D0Y8SB 4355631 Ki > 10000 nM T77365 D0YR1V 135457998 IC50 = 71 nM T77365 D0Z1WY 44447548 Ki > 100000 nM T77365 D0Z2QM 23562742 Ki = 12000 nM T77365 D0Z3XC 11185362 Ki = 255.3 nM T77365 D0Z7BC 44442164 Ki > 10000 nM T77365 D0Z8NC 16109435 Ki = 194 nM T77365 D0Z8VU 44572295 Ki = 390 nM T77365 D0ZD4M 834731 Ki = 2900 nM T77365 D0ZF8N 11196622 Ki > 1000 nM T77365 D0ZV1T 11371386 Ki = 381 nM T77365 D0ZW9L 11150373 Ki = 192 nM T81780 CD8Q1P 10432257 IC50 = 40000 nM T81780 CGD6Q1 44575998 IC50 = 17 ug.mL-1 T81780 CAX70H 70684035 IC50 = 35000 nM T81780 CUB35H 70694527 IC50 = 2400 nM T81780 D0Z8PX 24757913 IC50 = 29000 nM T78581 CZ63PR 16133811 Ki = 0.03 nM T78581 CP42JF 25180487 Ki = 1.9 nM T78581 C5VA6W 25180488 Ki = 25.5 nM T78581 CZ51CD 25180490 Ki = 3.3 nM T78581 C1IU8X 25180491 Ki = 0.9 nM T78581 C2WMX8 25180492 Ki = 25.5 nM T78581 CZ1N7I 25180493 Ki = 0.4 nM T78581 C3G8OJ 25180494 Ki = 6 nM T78581 CHRV59 25180496 Ki = 21.5 nM T78581 CVN29B 25180497 Ki = 41.5 nM T78581 C62QZX 25180498 Ki = 306.5 nM T78581 CK4J9W 44584852 IC50 = 0.079 nM T78581 C0GTZ7 44587983 Ki = 85 nM T78581 C20WUX 44587984 Ki = 3.5 nM T78581 C1TO0M 57390716 IC50 = 5480 nM T78581 CKE01G 57390718 IC50 = 6820 nM T78581 C32ETJ 57392517 IC50 = 5930 nM T78581 C7AT3L 57394236 IC50 = 4600 nM T78581 CY5D0W 57394237 IC50 = 5620 nM T78581 CJ39YQ 57394238 IC50 = 1300 nM T78581 CN0MS2 57394304 IC50 = 34860 nM T78581 COJ7T1 57395992 IC50 = 6770 nM T78581 CU6K8A 57395993 IC50 = 27500 nM T78581 CU93SZ 57395994 IC50 = 3900 nM T78581 CJZ65X 57395996 IC50 = 3840 nM T78581 CB70EI 57396058 IC50 = 8590 nM T78581 C7GK1B 57397798 IC50 = 3350 nM T78581 C2W0JH 57399456 IC50 = 12800 nM T78581 C2H3XW 57399457 IC50 = 6820 nM T78581 CZ9RD1 57399458 IC50 = 6320 nM T78581 CS27BV 57401220 IC50 = 6900 nM T78581 C8DS7R 57401221 IC50 = 5030 nM T78581 CT7PZ3 57401225 IC50 = 6780 nM T78581 C72GPE 57401226 IC50 = 3840 nM T78581 C4GJ3E 57401227 IC50 = 16010 nM T78581 CG1J8I 57401228 IC50 = 2820 nM T78581 CYR89Z 71508528 Ki = 3.8 nM T78581 CDJ2N3 71717271 Ki = 11700 nM T78581 C0O3CM 71720536 Ki = 37.5 nM T78581 D01LMH 25180489 Ki = 2.8 nM T78581 D02GOE 44563954 Ki = 1.4 nM T78581 D02JQP 24760995 Ki = 3.5 nM T78581 D03ECE 44563952 Ki = 0.7 nM T78581 D05GFD 44563953 Ki = 1.3 nM T78581 D06DWA 44563958 Ki = 0.5 nM T78581 D07NOJ 45104655 Ki = 11 nM T78581 D08FGR 24748735 Ki = 34200 nM T78581 D09SDZ 44587982 Ki = 0.5 nM T78581 D0DD3F 44563955 Ki = 2.6 nM T78581 D0EO5F 44563956 Ki = 3.5 nM T78581 D0H4DF 16132126 Ki = 0.03 nM T78581 D0H9QA 25180495 Ki = 387 nM T78581 D0PY7O 6324638 Ki = 870 nM T78581 D0Q3CB 16133821 Ki = 0.1 nM T78581 D0S4VO 45104657 Ki = 364.5 nM T78581 D0TF7R 44563951 Ki = 0.4 nM T78581 D0V7UG 45104656 Ki = 1.7 nM T78581 D0Z3QG 44563957 Ki = 4 nM T55986 C7NW5T 44555355 IC50 > 20 nM T55986 CIW0H6 50899478 IC50 > 20 nM T55986 C5QU2O 50899571 IC50 > 20 nM T55986 C8WD6E 50899573 IC50 > 20 nM T55986 C29AKS 118717990 IC50 > 20 nM T55986 CU4O3M 118718077 IC50 > 20 nM T55986 CS16DB 118718078 IC50 > 20 nM T55986 CK6E3L 118718085 IC50 > 20 nM T92403 D0N8QQ 151172 IC50 > 30000 nM T92403 D0V9RU 6433092 IC50 > 30000 nM T92403 CWC0M2 9925502 IC50 > 30000 nM T92403 CB0J1G 46174396 IC50 = 28 nM T92403 CJ68YT 58393461 IC50 = 0.2 nM T92403 CY9I6G 58393477 IC50 = 22 nM T92403 CAI83V 58393493 IC50 = 588 nM T92403 C65ORN 58393495 IC50 = 94 nM T92403 CC64UW 58393507 IC50 = 166 nM T92403 CU8P6Q 58393510 IC50 = 540 nM T92403 C4COR1 58393517 IC50 = 197 nM T92403 CP0D3T 58393548 IC50 = 118 nM T92403 C0ISF3 58393567 IC50 = 640 nM T92403 CE3ZR5 58393570 IC50 = 43 nM T92403 C2Z7GP 58393580 IC50 = 3520 nM T92403 CW05LJ 58393592 IC50 = 135 nM T92403 CP58EX 58393618 IC50 = 6680 nM T92403 CXAE04 58393620 IC50 = 168 nM T92403 CNW5T4 58393622 IC50 = 23 nM T92403 C2O9AB 58393629 IC50 = 4 nM T92403 CWU20N 58393632 IC50 = 411 nM T92403 CY6F0D 58393650 IC50 = 30 nM T92403 C7X8AL 58393659 IC50 = 345 nM T92403 CS7QM5 58393676 IC50 = 9520 nM T92403 C6L5WJ 58393694 IC50 = 2070 nM T92403 C0DSJ7 58393711 IC50 = 30 nM T92403 C4B0TS 58393722 IC50 = 11 nM T92403 CE9F2D 58393733 IC50 = 6055 nM T92403 CD24KR 58393739 IC50 = 272 nM T92403 C0J6DV 58393772 IC50 = 20 nM T92403 CF7U6N 58393782 IC50 = 17 nM T92403 CG8SJ7 58393792 IC50 = 4040 nM T92403 CID75X 58393839 IC50 = 48 nM T92403 C1P5ED 58393847 IC50 = 955 nM T92403 CUKP69 58393851 IC50 = 6 nM T92403 CVW3J5 58393864 IC50 = 64 nM T92403 CF39ET 58393876 IC50 = 1640 nM T92403 CG50XR 58393885 IC50 = 90 nM T92403 CC7LE9 58393895 IC50 = 93 nM T92403 CML4G7 58393897 IC50 = 1710 nM T92403 CSGL45 58393901 IC50 = 883 nM T92403 COD27G 58393915 IC50 = 23 nM T92403 CJ9P7S 58393925 IC50 = 78 nM T92403 CFM0W2 58393927 IC50 = 170 nM T92403 C84USG 58393938 IC50 = 241 nM T92403 CB6Y9V 58393939 IC50 = 737 nM T92403 CH90SQ 58393941 IC50 = 20 nM T92403 CHPD56 58393945 IC50 = 56 nM T92403 CQP93G 58393958 IC50 = 3490 nM T92403 C4TY9M 58394051 IC50 = 123 nM T92403 CBK90P 58394053 IC50 = 2960 nM T92403 CR8F2V 58394079 IC50 = 1530 nM T92403 CA2H5P 58394127 IC50 = 4500 nM T92403 C2O5AJ 58394134 IC50 = 384 nM T92403 C54QRX 58394136 IC50 = 34 nM T92403 CYW78T 58394137 IC50 = 572 nM T92403 CTCP38 58394149 IC50 = 540 nM T92403 C6SJH5 58394151 IC50 = 2 nM T92403 CD2YF7 58394180 IC50 = 2440 nM T92403 CT1RB3 67309779 IC50 = 4 nM T92403 CQ70DL 67311221 IC50 = 440 nM T92403 CX6YS0 117717369 IC50 = 4530 nM T92403 C4LZ8T 134133503 IC50 = 475 nM T92403 CYI93Q 134136642 IC50 = 438 nM T92403 CD8Z3Q 134147673 IC50 = 2770 nM T92403 CY54BL 134152502 IC50 = 123 nM T92403 CKU7X4 134152809 IC50 = 330 nM T92403 CBPN64 134154817 IC50 = 281 nM T92403 CTX8Q6 134155895 IC50 = 650 nM T92403 C9LI1Z 134156817 IC50 = 500 nM T20514 CYZE76 459456 IC50 = 511000 nM T20514 CZ7UE4 2735808 IC50 = 85300 nM T20514 C8OX1T 2757170 IC50 = 99700 nM T20514 CT9ZW4 3307674 IC50 = 500000 nM T20514 C80SHO 4913063 IC50 = 500000 nM T20514 CK8GS4 28547001 IC50 = 222000 nM T20514 CM0HF7 29296769 IC50 = 156000 nM T20514 C2D1QC 29559943 IC50 = 213000 nM T20514 CV4DF0 42817381 IC50 = 740000 nM T20514 CW4YN6 50956414 IC50 = 119000 nM T20514 CDPX96 50965913 IC50 > 1000000 nM T20514 C8QKR9 71044558 IC50 = 145000 nM T20514 CL3GB6 83413959 IC50 = 173000 nM T20514 C8J2KR 90643851 IC50 = 500000 nM T20514 C51VFU 90643852 IC50 = 197000 nM T20514 CJS5C4 90643853 IC50 = 500000 nM T20514 CL9OM3 90643854 IC50 = 500000 nM T20514 C14SPD 90643855 IC50 = 500000 nM T20514 C7CZ0E 90643856 IC50 = 637000 nM T20514 CG5NS4 21158826 Ki = 200000000 nM T81311 D01FYA 9549213 IC50 = 26 nM T81311 D05BYA 135539077 Ki = 4 nM T81311 D05HWN 16736529 Ki = 176 nM T81311 D0F3NF 67501411 Ki > 50000 nM T81311 CYQP95 11198704 IC50 = 350 nM T81311 CO3F6K 11221466 IC50 = 1130 nM T81311 CH4B2Z 11223683 IC50 = 170 nM T81311 CBZS48 11302159 IC50 = 1630 nM T81311 CDJX31 11326407 IC50 = 530 nM T81311 C2ZCY3 11336657 IC50 = 11450 nM T81311 CIRH67 11349446 IC50 = 120 nM T81311 CUO6Q7 11393625 IC50 = 29400 nM T81311 CXN76P 11406285 IC50 = 260 nM T81311 CP3Z4O 11407267 IC50 = 500 nM T81311 CP90LC 11427896 IC50 = 1500 nM T81311 CR9IQ7 11450570 IC50 = 1140 nM T81311 C8VZQ6 11463506 IC50 = 1400 nM T81311 CI53RD 11473241 IC50 = 6200 nM T81311 C9IY1M 11517212 Ki = 61 nM T81311 C79VTC 11773074 IC50 = 34500 nM T81311 COBM26 25073055 IC50 = 101 nM T81311 CZ7XQ5 60165612 IC50 = 1200 nM T81311 CAU06M 66576834 IC50 = 265 nM T81311 CV8B0R 67495834 Ki = 375 nM T81311 CIG6P3 71660550 IC50 = 2100 nM T81311 C79AGJ 71660551 IC50 = 220 nM T81311 C9CW5M 73437615 Ki > 10000 nM T81311 CUD54E 73437616 Ki > 10000 nM T81311 CS0PB2 76324772 Ki = 2650 nM T81311 CJ3Q4H 90654630 Ki > 10000 nM T81311 CG8S1L 90654631 Ki = 2400 nM T81311 CDIY85 90654632 Ki > 10000 nM T81311 CV9YA4 90654633 Ki > 10000 nM T81311 CRH14E 90654634 Ki > 10000 nM T81311 C26WSJ 90654635 Ki > 10000 nM T81311 CXLQ38 90654636 Ki > 10000 nM T81311 C9F5UB 90654637 Ki > 10000 nM T81311 CZ2MP4 90654638 Ki > 10000 nM T81311 C17RWB 90654639 Ki > 10000 nM T81311 C7X8WK 90654640 Ki = 4400 nM T81311 CJ2ZM3 90654641 Ki = 1100 nM T81311 C21FPZ 90654642 Ki = 580 nM T81311 C9ZTU1 90654643 Ki = 2800 nM T81311 CTB60Y 90654644 Ki > 10000 nM T81311 C81JGB 90654645 Ki = 420 nM T81311 CKM2W0 90654646 Ki = 3200 nM T81311 CS8U1X 90654647 Ki > 10000 nM T81311 CUE4I6 90654648 Ki = 3700 nM T81311 CM5JP8 90654649 Ki = 620 nM T81311 CH8FD0 90654650 Ki = 2900 nM T81311 C5DP2C 90654651 Ki = 840 nM T81311 CU87TN 90654652 Ki > 10000 nM T81311 C4PJ1V 90654653 Ki > 10000 nM T81311 C2TYR0 90654654 Ki > 10000 nM T81311 C6SI7L 90654655 Ki > 10000 nM T81311 CG2JK7 90654656 Ki > 10000 nM T81311 CBWT05 90654657 Ki > 10000 nM T81311 C2TLY1 90654659 Ki > 10000 nM T81311 C3R1DJ 90654660 Ki > 10000 nM T81311 CT1QI5 90654661 Ki > 10000 nM T81311 CU8Q1V 90654662 Ki > 10000 nM T81311 CS42OM 90654663 Ki > 10000 nM T81311 C7M8TA 90654664 Ki > 10000 nM T81311 C1H5WC 90654665 Ki > 10000 nM T81311 CUVD12 117889758 IC50 = 4700 nM T81311 CUTV54 117889766 IC50 = 287 nM T81311 CIBF07 117889785 IC50 = 500 nM T81311 CW8J2A 117889863 IC50 = 2480 nM T81311 CP0VL5 117889908 IC50 = 5400 nM T81311 C0GZD8 117889984 IC50 = 700 nM T81311 CGM51T 117890044 IC50 > 5000 nM T81311 C37QWO 117890084 IC50 = 1648 nM T81311 C1APC8 117890111 IC50 = 430 nM T81311 CZ4EN5 117890133 IC50 > 2500 nM T81311 CO2R1E 117890146 IC50 = 502 nM T81311 CE69YR 117890174 IC50 > 5000 nM T81311 C3C6KX 117890187 IC50 = 1900 nM T81311 CX6V7Q 117890195 IC50 = 560 nM T81311 C4MQ8T 117890212 IC50 = 290 nM T81311 CG53QV 117890216 IC50 = 410 nM T81311 CZ45SB 117890250 IC50 = 340 nM T81311 CLH49C 117890268 IC50 = 665 nM T81311 CLHP30 117890308 IC50 = 2740 nM T81311 CQK30X 117890321 IC50 = 7730 nM T81311 CPWS97 117890346 IC50 = 14300 nM T81311 C1HK7L 117890351 IC50 = 390 nM T81311 CO25TC 117890352 IC50 = 5100 nM T81311 CA15DJ 117890354 IC50 = 429 nM T81311 CTV53C 117890368 IC50 = 695 nM T81311 CQCT02 117890387 IC50 = 920 nM T81311 CQ20HF 117890473 IC50 = 3440 nM T81311 C3R9DT 117890494 IC50 = 240 nM T81311 CRYX09 117890515 IC50 = 1080 nM T81311 CKE49U 118737375 IC50 = 5800 nM T81311 C84YNW 118737376 IC50 = 800 nM T81311 CKB9N5 118737377 IC50 = 390 nM T81311 C1ZSK4 118737378 IC50 = 5000 nM T81311 C2SRX9 136198647 IC50 > 100000 nM T81311 CEX34H 136198648 IC50 = 100000 nM T81311 CN0XY9 136198649 IC50 > 100000 nM T81311 CP79HX 136198650 IC50 = 2080 nM T81311 CR3LD9 136198651 IC50 = 20000 nM T81311 CN83ZX 136198652 IC50 > 25000 nM T81311 CEWC75 136198653 IC50 = 2430 nM T81311 C2NOH9 136236968 IC50 = 11770 nM T81311 CTCO28 136934953 IC50 = 100000 nM T81311 CMZ90X 136934954 IC50 > 100000 nM T81311 CW40ER 136934955 IC50 > 100000 nM T81311 CKS79P 136934956 IC50 > 100000 nM T81311 CA4OC9 136934957 IC50 = 2370 nM T81311 CI8FR0 136934958 IC50 = 11770 nM T81311 C5VIG4 136934959 IC50 > 100000 nM T81311 C2YZ6E 136934960 IC50 = 35300 nM T81311 C6B4DY 136934961 IC50 > 100000 nM T81311 D0K0TJ 24772860 Ki = 484 nM T60213 D0E3TC 44259 IC50 = 1100 nM T60213 D0S1XX 134821691 IC50 = 193 nM T60213 CPQ31L 25195294 IC50 = 3845 nM T60213 C91FTP 57339386 IC50 = 24 nM T60213 CIP7B1 60182373 IC50 = 59 nM T60213 CQ6KV9 60182388 IC50 = 695 nM T60213 CV63UL 67240318 IC50 > 10000 nM T60213 CPT0V7 138454752 IC50 > 10000 nM T60213 C2MD1Q 155513187 IC50 > 10000 nM T60213 D05NEC 60182364 IC50 = 2360 nM T60213 D0F2MP 60182389 IC50 = 3640 nM T60213 D0PP6Y 60182393 IC50 = 15.9 nM T60213 D0Y0BK 11524144 IC50 = 74 nM T85574 D00JAU 3749 IC50 = 3 nM T85574 D0K0AT 6324663 IC50 = 0.066 nM T85574 D08AWI 11430856 Ki > 2000 nM T85574 D0F2HA 132562 IC50 = 31 nM T85574 D0GS7N 183134 IC50 = 0.3 nM T85574 D0Y8PH 9828975 IC50 = 3.8 nM T85574 CTCP47 130762 IC50 = 230 nM T85574 C81FHI 171012 IC50 = 0.45 nM T85574 CBEW80 187067 IC50 = 2 nM T85574 CD10GC 190830 IC50 = 0.08 nM T85574 C6UO1X 3036053 IC50 = 1 nM T85574 CN9A2Q 4110026 IC50 = 2300 nM T85574 CKWP24 4286584 IC50 = 96 nM T85574 C20VPT 5249743 IC50 = 22 nM T85574 CNDM64 5748380 IC50 = 5.8 nM T85574 CQJ76K 9805248 IC50 = 3.48 nM T85574 CY6ZC3 9806554 IC50 = 1 nM T85574 CH2FD7 9809280 IC50 = 920 nM T85574 C2YCP6 9871452 IC50 = 0.4 nM T85574 CM3N8S 9887844 IC50 = 5 nM T85574 CEO03B 9889557 IC50 = 17 nM T85574 C5YT2C 9892554 IC50 = 0.2 nM T85574 CG9I2F 9916833 IC50 = 1.7 nM T85574 CJF49M 9960721 IC50 = 350 nM T85574 CRL65O 9979771 IC50 = 44 nM T85574 C78POU 9981102 IC50 = 40 nM T85574 C9DAJ6 9984181 IC50 = 10 nM T85574 C96IMW 9985923 IC50 = 4 nM T85574 C8BUA4 10001550 IC50 = 2 nM T85574 CFTL14 10004646 IC50 = 18 nM T85574 C0TNH6 10005512 IC50 = 0.7 nM T85574 CYF76W 10005890 IC50 = 28 nM T85574 CEX02H 10006024 IC50 = 0.1 nM T85574 CA8H2D 10025443 IC50 = 0.8 nM T85574 C0C5FR 10027175 IC50 > 100 nM T85574 C06TYP 10028209 IC50 = 0.4 nM T85574 CWL2S3 10030062 IC50 = 9.2 nM T85574 CS0BA9 10030110 IC50 = 2.9 nM T85574 COR34E 10030704 IC50 = 2 nM T85574 CDH6Y0 10048770 IC50 = 32 nM T85574 CHDB84 10049809 IC50 = 35 nM T85574 CG8W2R 10050932 IC50 = 0.3 nM T85574 CN8GS2 10054827 IC50 = 7 nM T85574 CC5GW1 10075811 IC50 = 370 nM T85574 C46RWQ 10076233 IC50 = 3 nM T85574 CNQ97X 10079601 IC50 = 0.21 nM T85574 CME6A5 10093043 IC50 = 0.7 nM T85574 CP0I6R 10099052 IC50 = 3 nM T85574 C2Z4UC 10099291 IC50 = 1 nM T85574 CL31NR 10168097 IC50 = 2 nM T85574 CM1X7P 10252636 IC50 = 0.7 nM T85574 CKX80Y 10254585 IC50 = 14 nM T85574 CV8Q3T 10256452 IC50 = 2 nM T85574 CUK72W 10256602 IC50 = 5.3 nM T85574 CE0Q7N 10257189 IC50 = 97 nM T85574 C8KAP3 10257584 IC50 > 100 nM T85574 CNC45L 10323474 IC50 = 0.5 nM T85574 CH21JQ 10324361 IC50 > 100 nM T85574 CHJ4G0 10325267 IC50 = 290 nM T85574 CW7K4Z 10342301 IC50 = 28 nM T85574 C4XZO9 10343090 IC50 = 30 nM T85574 CN2SW3 10346824 IC50 = 120 nM T85574 CF57JW 10348832 IC50 = 460 nM T85574 CWZ9N7 10367792 IC50 = 28 nM T85574 CVD5W6 10369701 IC50 = 490 nM T85574 CX5S6U 10369826 IC50 = 2 nM T85574 CSUH47 10369867 IC50 = 21 nM T85574 CX8MP7 10370006 IC50 = 0.1 nM T85574 C8EBV1 10391038 IC50 = 460 nM T85574 C5E8WI 10392378 IC50 = 2.6 nM T85574 C70JVE 10393016 IC50 = 12 nM T85574 C9VR4Z 10393086 IC50 = 500 nM T85574 CL9U5B 10404658 IC50 = 9400 nM T85574 CJ73AH 10414201 IC50 = 2400 nM T85574 C9MRQ6 10414273 IC50 > 100 nM T85574 C1XST2 10414338 IC50 = 13 nM T85574 C42BDV 10414470 IC50 = 40 nM T85574 C1BS9U 10414660 IC50 = 1900 nM T85574 C6DYJ7 10430907 IC50 = 2 nM T85574 CZ4M9S 10436366 IC50 = 0.3 nM T85574 CQAM96 10437372 IC50 = 4 nM T85574 CQV4W0 10438031 IC50 = 0.3 nM T85574 CXA9I8 10456587 IC50 = 0.6 nM T85574 CLT9Y5 10460419 IC50 = 0.8 nM T85574 C5IFH8 10478294 IC50 = 74 nM T85574 CEX94Z 10482431 IC50 = 90 nM T85574 C1M6NL 10482664 IC50 = 10 nM T85574 C3XK5L 10504330 IC50 = 89 nM T85574 C0GO1E 10674630 IC50 = 28 nM T85574 CZRC03 10697700 IC50 = 15 nM T85574 CS2U9K 10697829 IC50 = 52 nM T85574 C3BYA7 10744859 IC50 = 26 nM T85574 CV2E4Z 11476710 IC50 = 3 nM T85574 C7XH5K 11755602 IC50 = 0.2 nM T85574 CJVM73 11756968 IC50 = 0.2 nM T85574 CZ2C1H 11801362 IC50 = 38 nM T85574 C1RT7B 14950512 IC50 = 14 nM T85574 C8S3KM 14962839 IC50 = 7 nM T85574 CJ26VO 14962840 IC50 > 100 nM T85574 C3XJ5E 14962841 IC50 = 400 nM T85574 C57MBD 14962842 IC50 = 5400 nM T85574 CC7TD9 14962843 IC50 = 52 nM T85574 CKZ5I2 14962844 IC50 = 4 nM T85574 CAPM52 14962845 IC50 = 330 nM T85574 CF21BT 14962846 IC50 = 5.4 nM T85574 C6YAR2 14962847 IC50 = 1500 nM T85574 C5E7AU 14962848 IC50 = 3500 nM T85574 CL5PD7 14962849 IC50 = 780 nM T85574 CE5P3J 14962850 IC50 = 2200 nM T85574 CGP82M 14962851 IC50 = 2400 nM T85574 C2FZ3A 14962853 IC50 = 57 nM T85574 CET31Z 14962854 IC50 = 73 nM T85574 C1LJF6 14962855 IC50 = 19 nM T85574 C8I6QU 14962856 IC50 = 150 nM T85574 C5F3AR 14962857 IC50 = 2.35 nM T85574 C58HDA 14962858 IC50 > 100 nM T85574 CT89EB 14962859 IC50 = 4.5 nM T85574 C20YQM 14962860 IC50 > 100 nM T85574 CHY9X3 14962861 IC50 = 82 nM T85574 C6Z7NT 14962862 IC50 = 9 nM T85574 C6KA8M 14962863 IC50 > 100 nM T85574 CXZ6Q4 14962866 IC50 = 71 nM T85574 C8K3MH 14962867 IC50 = 39 nM T85574 CH6PF0 14962868 IC50 = 2.9 nM T85574 C1R0FV 14962869 IC50 = 2.6 nM T85574 CN3RK1 14962873 IC50 = 34 nM T85574 CSB3X5 14962875 IC50 = 21 nM T85574 CM75EG 14962876 IC50 > 100 nM T85574 CG52CA 14962877 IC50 = 18 nM T85574 CJ8MP7 14962878 IC50 = 430 nM T85574 CCL31T 14962879 IC50 = 3.3 nM T85574 CWL32U 14987298 IC50 = 1800 nM T85574 CK6UD7 15069293 IC50 = 140000 nM T85574 CGQ6N0 15076143 IC50 = 8 nM T85574 CTS79R 15076144 IC50 = 2 nM T85574 C7P9ML 15076145 IC50 = 0.5 nM T85574 CTU4X8 15076146 IC50 = 0.3 nM T85574 CCZ83E 15129910 IC50 = 7400 nM T85574 C42MSA 15129911 IC50 = 51000 nM T85574 CD5T2J 15129918 IC50 = 4900 nM T85574 C8IRL0 15129919 IC50 = 7100 nM T85574 CG87PK 15129920 IC50 = 11000 nM T85574 CD9W8Y 15129921 IC50 = 640 nM T85574 C1VZR5 15129926 IC50 = 8500 nM T85574 C0B6UQ 15129928 IC50 = 1600 nM T85574 C9IPK8 15129933 IC50 = 860 nM T85574 C3UHL2 15129934 IC50 = 3700 nM T85574 C8PLG7 15129935 IC50 = 18000 nM T85574 CVJ63Z 15129936 IC50 = 1800 nM T85574 CQ6XY1 15129937 IC50 = 5400 nM T85574 C57MLE 15129938 IC50 = 3900 nM T85574 CW0Y9Z 15129939 IC50 = 12000 nM T85574 C2TP3Y 15690078 IC50 > 15000 nM T85574 C4VA7E 15690082 IC50 > 15000 nM T85574 CURS43 15690085 IC50 > 15000 nM T85574 CA30YX 19012962 IC50 = 220 nM T85574 C5Z6NF 19742867 IC50 = 3.83 nM T85574 CKJ5W0 19742873 IC50 = 2.64 nM T85574 CEK56J 19742883 IC50 = 7.58 nM T85574 C3AD8M 19742889 IC50 = 6.65 nM T85574 C54PXI 19742895 IC50 = 8.03 nM T85574 CA6EJ4 19742907 IC50 = 24.9 nM T85574 CI2Z1D 19815363 IC50 = 400 nM T85574 C03NRE 20604663 IC50 = 10000 nM T85574 C3KSI1 21831269 IC50 = 6.8 nM T85574 C4IXZ1 44209569 IC50 = 22 nM T85574 CR28CF 44264673 IC50 = 2130 nM T85574 CVIC87 44264684 IC50 = 10000 nM T85574 CH84VM 44264772 IC50 = 100000 nM T85574 C7IRH2 44264838 IC50 = 255 nM T85574 CRMV49 44281252 IC50 = 6.21 nM T85574 C2EW6X 44281532 IC50 = 26.4 nM T85574 C4O3FZ 44284136 IC50 = 280 nM T85574 CY0S7U 44289773 IC50 = 0.2 nM T85574 C7EAB1 44312598 IC50 = 4.8 nM T85574 CY5U8K 44312630 IC50 > 100 nM T85574 C9FEA1 44317243 IC50 = 7 nM T85574 CEC24I 44317309 IC50 > 15000 nM T85574 CMKZ39 44321474 IC50 = 42 nM T85574 CE6WJ9 44321475 IC50 = 10.6 nM T85574 CY35QF 44321476 IC50 = 5.8 nM T85574 CNS63J 44321486 IC50 = 2.5 nM T85574 C49WTZ 44321736 IC50 = 9 nM T85574 CCQ63Z 44321846 IC50 = 5.4 nM T85574 CF04UN 44321848 IC50 = 28 nM T85574 CGM47N 44321870 IC50 = 55 nM T85574 CIE63T 44321871 IC50 = 23 nM T85574 C24CKI 44321872 IC50 = 3.4 nM T85574 C5YO7D 44321894 IC50 = 14.3 nM T85574 C6JGW7 44321895 IC50 = 367 nM T85574 C8NX0R 44321896 IC50 = 2200 nM T85574 C2V8UT 44321897 IC50 = 9.5 nM T85574 C1XJY3 44322030 IC50 = 44 nM T85574 COC09T 44322031 IC50 = 20 nM T85574 C8U0XZ 44322032 IC50 = 7.8 nM T85574 CD9O5M 44322057 IC50 = 850 nM T85574 C1I3LW 44322058 IC50 = 170 nM T85574 C5S0VM 44322059 IC50 = 17 nM T85574 CZI95P 44322079 IC50 = 190 nM T85574 CL5OH1 44322094 IC50 = 17 nM T85574 C8X0EZ 44322139 IC50 = 220 nM T85574 CK3Y2E 44322267 IC50 = 1.3 nM T85574 C9JUQ1 44322268 IC50 = 7 nM T85574 CU1V0F 44330457 IC50 = 6 nM T85574 CVXW61 44382465 IC50 = 15000 nM T85574 CVH2U1 44460414 IC50 > 10000 nM T85574 C8A7XU 44460431 IC50 = 3600 nM T85574 CCT7S2 44461082 IC50 > 10000 nM T85574 C75RNT 44461110 IC50 = 5000 nM T85574 CE4X9Q 45263060 IC50 = 5600 nM T85574 CC6S4W 73348444 IC50 = 0.2 nM T85574 C14LGZ 73351521 IC50 = 330 nM T85574 CIEG15 155527749 IC50 = 200 nM T85574 D0D1FT 108185 IC50 = 1.8 nM T15795 D08HQK 5411 IC50 = 668000 nM T15795 D09RHQ 175805 IC50 = 53000 nM T15795 D0A0FL 2474 IC50 = 41000 nM T15795 D0G7DJ 37497 IC50 = 39000 nM T15795 D0J2KV 4932 IC50 = 5100 nM T15795 D0WO8W 4062 IC50 = 709000 nM T15795 D0X0RI 4178 IC50 = 97300 nM T15795 D0X4RN 3676 IC50 = 222000 nM T15795 D07LWK 9811357 IC50 = 600 nM T15795 CPDW86 252604 IC50 = 240 nM T15795 CMSU69 738674 IC50 = 45 nM T15795 CSMB29 759456 IC50 = 30 nM T15795 C5CK1Q 825574 IC50 = 140 nM T15795 CYX02K 825799 IC50 = 27 nM T15795 CQ62XP 825801 IC50 = 37 nM T15795 CH30JL 869662 IC50 = 330 nM T15795 CDM4O2 902575 IC50 = 29 nM T15795 C3FW4S 1019323 IC50 = 10 nM T15795 C16DWN 1085239 IC50 = 190 nM T15795 C7GE8N 1154076 IC50 = 500 nM T15795 C2AGB0 1248054 IC50 = 1290 nM T15795 CQ3O0J 1376748 IC50 > 3000 nM T15795 C75PBL 1377831 IC50 = 73 nM T15795 CEY81D 2840308 IC50 = 220 nM T15795 C8TSE4 3097786 IC50 > 3000 nM T15795 CMU4F3 3396992 IC50 = 91 nM T15795 C4HMG0 3658964 IC50 = 310 nM T15795 CH9TO2 3745727 IC50 = 3200 nM T15795 C95QEX 9540179 IC50 = 52 nM T15795 C05GSU 9825796 IC50 = 1050 nM T15795 CGBE91 9827303 IC50 = 7 nM T15795 C0HXS3 10236329 IC50 = 51000 nM T15795 C35GHD 15812076 IC50 > 3000 nM T15795 C6XP3O 17234805 IC50 = 100 nM T15795 CFS36C 17234818 IC50 > 3000 nM T15795 C97WQE 17234824 IC50 > 3000 nM T15795 C8A2UI 17234870 IC50 = 250 nM T15795 CD51EA 17744755 IC50 = 79 nM T15795 CB7Z6S 22006193 IC50 = 350 nM T15795 C6RY9W 31520618 IC50 = 5 nM T15795 C2SOY1 46785920 IC50 = 4 nM T15795 CL2A8W 46785922 IC50 = 25 nM T15795 CFZ75O 46880148 IC50 = 3 nM T15795 C9N6GZ 49793697 IC50 = 96700 nM T15795 CJ8UN9 49793859 IC50 = 83500 nM T15795 CT2BL8 49842926 IC50 = 160 nM T15795 CP27XZ 49852186 IC50 = 1300 nM T15795 CLW51Q 49852187 IC50 > 3000 nM T15795 C0NK5Z 49852188 IC50 = 23 nM T15795 C4UBV9 49852189 IC50 = 31 nM T15795 CV10JQ 49852190 IC50 = 260 nM T15795 CL59YO 49852191 IC50 = 95 nM T15795 C7ZUF5 49852192 IC50 = 10 nM T15795 CSVZ76 49852193 IC50 = 800 nM T15795 C6KX1V 49852195 IC50 = 14 nM T15795 C07TWM 49867945 IC50 = 160 nM T15795 C5P4AK 49867946 IC50 = 130 nM T15795 CA2P0D 49867948 IC50 = 150 nM T15795 CFE80H 49867949 IC50 = 86 nM T15795 C0Z8FV 49867950 IC50 = 150 nM T15795 CODR75 50919318 IC50 = 330 nM T15795 CPF0H1 50919319 IC50 = 9 nM T15795 C13IBD 50919320 IC50 = 29 nM T15795 C1O6QP 51049782 IC50 = 4 nM T15795 CVT26J 51049785 IC50 = 2 nM T15795 C4VQT0 51049787 IC50 = 7 nM T15795 C7PU3H 51358807 IC50 = 10 nM T15795 C9WS3Z 53301908 IC50 = 11 nM T15795 C9D7AH 53301913 IC50 = 1 nM T15795 C48QEY 53464059 IC50 = 300 nM T15795 CRM42J 58892059 IC50 = 220 nM T15795 C3NS2C 118708433 IC50 = 150 nM T15795 C3XZY7 118708434 IC50 = 210 nM T15795 C0AM1J 118708435 IC50 = 180 nM T15795 D07VWP 656730 IC50 = 200 nM T15795 D0A9PS 5281969 IC50 = 3000 nM T15795 D0I4YK 6321351 IC50 = 100 nM T74864 C79IRE 71620755 IC50 = 360 nM T74864 C7PI9C 71620756 IC50 = 360 nM T74864 CGD70V 71620759 IC50 = 360 nM T74864 CX85HD 71621073 IC50 = 360 nM T74864 CZB46R 71621227 IC50 = 360 nM T74864 CNP1U5 86574151 IC50 = 360 nM T74864 C2LM9W 127026354 IC50 = 30 nM T74864 CRD02W 127026355 IC50 = 280 nM T74864 C6KE3B 127026667 IC50 = 80 nM T74864 CE2PX6 127026668 IC50 = 30 nM T74864 C7VP6A 127026669 IC50 = 10 nM T74864 C1IF8B 127028921 IC50 = 70 nM T74864 C5ZK6J 127029217 IC50 = 50 nM T74864 CZ3DS8 127029218 IC50 = 40 nM T74864 CMR68I 127029233 IC50 = 1 nM T74864 C7ZHE4 127029234 IC50 = 10 nM T40492 D09ZZW 503536 IC50 = 1500 nM T40492 C6IQV0 482174 IC50 = 5700 nM T40492 CY61LO 487910 IC50 = 1700 nM T40492 C6K5JV 487911 IC50 = 16000 nM T40492 C3J5VH 487912 IC50 = 1000 nM T40492 CZNK70 487918 IC50 = 330 nM T40492 CDN3F2 487919 IC50 = 1630 nM T40492 CT76XW 487920 IC50 = 2100 nM T40492 CVA82G 487921 IC50 = 460 nM T40492 CBR46W 487922 IC50 = 1400 nM T40492 CAJ64Q 490750 IC50 < 1000 nM T40492 CMO49H 491114 IC50 = 4300 nM T40492 COB17R 492544 IC50 > 50000 nM T40492 C68MZE 492548 IC50 > 100000 nM T40492 C4JO9E 492549 IC50 = 3280 nM T40492 C1JEY2 492550 IC50 = 300 nM T40492 CRML27 492552 IC50 = 380 nM T40492 C84QRW 493418 IC50 = 5700 nM T40492 CY1WF7 497453 IC50 = 3000 nM T40492 C43PXV 503499 IC50 = 2400 nM T40492 C2BSI5 503516 IC50 = 14000 nM T40492 CFRT87 503517 IC50 = 5400 nM T40492 C3JB0U 503520 IC50 = 13000 nM T40492 CA72XJ 503521 IC50 = 5200 nM T40492 CF14KO 503522 IC50 = 7400 nM T40492 CH18YP 503523 IC50 = 4600 nM T40492 CG6T1D 503524 IC50 = 4100 nM T40492 CLY7T8 503525 IC50 = 750 nM T40492 C37MIA 503526 IC50 = 1000 nM T40492 C8U2AD 503527 IC50 = 12000 nM T40492 CO6R4G 503528 IC50 = 2000 nM T40492 CHA5F8 503529 IC50 > 50000 nM T40492 C41DVG 503530 IC50 = 21000 nM T40492 C5XRJ6 503531 IC50 = 1200 nM T40492 CI1V6W 503532 IC50 > 50000 nM T40492 C84DXH 503533 IC50 = 1400 nM T40492 C7R3CM 503534 IC50 = 2000 nM T40492 CCMU16 503535 IC50 = 3000 nM T40492 C1E4IO 504181 IC50 = 2700 nM T40492 CEJ6U1 504182 IC50 = 1800 nM T40492 CZDS90 504183 IC50 = 1600 nM T40492 C04ONL 504184 IC50 = 2200 nM T40492 C65XPH 504185 IC50 = 11000 nM T40492 CRZN68 504186 IC50 = 42000 nM T40492 CK8CA2 504187 IC50 > 60000 nM T40492 C01MYV 504188 IC50 = 5800 nM T40492 C4C5WD 504189 IC50 = 4300 nM T40492 CIB52E 504190 IC50 = 230 nM T40492 CQ6L1G 504191 IC50 = 12000 nM T40492 C4CW5A 504192 IC50 > 60000 nM T40492 C09ACU 504193 IC50 > 60000 nM T40492 C7T0AD 504194 IC50 = 1300 nM T40492 C7VZY1 504195 IC50 > 60000 nM T40492 CU4EK0 504196 IC50 = 3600 nM T40492 COUS53 504197 IC50 = 5300 nM T40492 CTE3B4 504198 IC50 = 7700 nM T40492 CT81MP 504676 IC50 = 3500 nM T40492 C9FI5K 504680 IC50 = 10600 nM T40492 C8IFN4 504681 IC50 = 31000 nM T40492 CV6OY3 506523 IC50 = 1400 nM T40492 CQX7S4 506524 IC50 = 390 nM T40492 CXD73I 506525 IC50 = 1800 nM T40492 C6ANI5 506528 IC50 = 9000 nM T40492 CRU30I 507613 IC50 = 900 nM T40492 CI8SQ4 511361 IC50 > 50000 nM T40492 C02LPN 511362 IC50 = 30000 nM T40492 CJIW67 511363 IC50 = 13000 nM T40492 C3KG1M 511364 IC50 = 43000 nM T40492 CU85HK 511365 IC50 = 10700 nM T40492 C20EKN 511366 IC50 = 5900 nM T40492 C3FX8J 511367 IC50 = 31000 nM T40492 C4DEY1 511368 IC50 = 3700 nM T40492 CC2J9M 511369 IC50 = 5600 nM T40492 CIU5M2 511370 IC50 = 11000 nM T40492 C5CG4I 511371 IC50 = 5000 nM T40492 CTO87P 511372 IC50 = 2700 nM T40492 C5BJ6S 511373 IC50 = 26000 nM T40492 CDWB40 511374 IC50 = 15000 nM T40492 CDH29C 511375 IC50 = 31000 nM T40492 C8ZJD7 511376 IC50 = 31000 nM T40492 CJ56OH 513150 IC50 < 10000 nM T40492 C5BN4U 513891 IC50 = 12000 nM T40492 CVI54C 657065 IC50 = 1200 nM T40492 CUC54L 3008068 IC50 = 5000 nM T40492 CJ5NO6 3008069 IC50 = 34000 nM T40492 CQO9Y3 3008070 IC50 > 32000 nM T40492 CXM1K9 3008071 IC50 > 50000 nM T40492 CJ2NY3 3008418 IC50 = 20000 nM T40492 CIJ2T0 3008419 IC50 > 50000 nM T40492 CWD1X0 3008420 IC50 = 14000 nM T40492 C4K2JP 3008421 IC50 > 50000 nM T40492 CAN83S 3008422 IC50 = 13000 nM T40492 CMDQ27 4468931 IC50 = 1800 nM T40492 CK9WY1 5278824 IC50 = 100 nM T40492 C5MEQ4 5278825 IC50 = 110 nM T40492 C1F0AN 5278826 IC50 = 45 nM T40492 CV0O6S 5482516 IC50 = 15600 nM T40492 CEM30Z 5483089 IC50 = 8900 nM T40492 CJL21S 9853197 IC50 = 60 nM T40492 CJW4M9 9917616 IC50 = 11000 nM T40492 C39ZBC 10207572 IC50 = 30000 nM T40492 CGA86Z 10259200 IC50 = 12000 nM T40492 CJ46UK 10439772 IC50 = 420 nM T40492 COM8C5 21148125 IC50 = 16000 nM T40492 C1TW3V 22209806 IC50 > 50000 nM T40492 C8GVX3 22209808 IC50 > 50000 nM T40492 C6AS7E 22209811 IC50 = 3300 nM T40492 CLW13P 22209812 IC50 = 1700 nM T40492 C1TA6Z 22209813 IC50 = 440 nM T40492 CGUC83 22210989 IC50 = 58000 nM T40492 CV97ER 22210996 IC50 = 18000 nM T40492 C2BA1K 22211000 IC50 = 27000 nM T40492 C78AKX 22211010 IC50 > 100000 nM T40492 CL7M9B 22211011 IC50 = 32000 nM T40492 C1L8TE 22211012 IC50 = 18000 nM T40492 C0NYS5 22211016 IC50 = 50000 nM T40492 C67QJW 22211018 IC50 > 100000 nM T40492 CV9S2O 22211019 IC50 = 13000 nM T40492 C4UB6Q 22211020 IC50 = 14000 nM T40492 CBUV46 22211021 IC50 = 62000 nM T40492 CS9B7N 22211022 IC50 > 100000 nM T40492 CK81WO 25078062 IC50 = 3400 nM T40492 CYDW71 44268661 IC50 > 60000 nM T40492 C6S3AT 44268682 IC50 > 60000 nM T40492 CDJ0X4 44308299 IC50 > 100000 nM T40492 CIO1C2 44308345 IC50 > 100000 nM T40492 CX14BI 44308422 IC50 > 100000 nM T40492 CE3PS8 44308752 IC50 = 34000 nM T40492 CK2P5O 44375061 IC50 > 50000 nM T40492 C4CVW1 44375110 IC50 > 50000 nM T40492 C72KUL 44375154 IC50 = 9400 nM T40492 C1SBO9 44375192 IC50 > 50000 nM T40492 C42GUE 44375229 IC50 = 5300 nM T40492 CX76FI 44388198 IC50 = 350 nM T40492 CVW6O4 44399745 IC50 = 79432.82 nM T40492 CDRP83 44399750 IC50 = 50118.72 nM T40492 CW6NY8 44399751 IC50 = 5011.87 nM T40492 CM5W8Q 44399752 IC50 = 6309.57 nM T40492 C34WSP 44399753 IC50 = 10000 nM T40492 CE0T1O 44399754 IC50 = 1995.26 nM T40492 CT86CR 44399784 IC50 = 25118.86 nM T40492 C6GWS9 44399837 IC50 = 31622.78 nM T40492 C4AI1T 44399861 IC50 = 100000 nM T40492 CTX79F 44399866 IC50 = 25118.86 nM T40492 CP4KB7 44399867 IC50 = 794.33 nM T40492 C0WRU5 44399868 IC50 = 15848.93 nM T40492 C8JP2A 44399889 IC50 = 50118.72 nM T40492 CO4H3V 44399938 IC50 = 10000 nM T40492 CYH7F9 44399975 IC50 = 6309.57 nM T40492 CZRF38 44399976 IC50 = 6309.57 nM T40492 CATH48 44399977 IC50 = 6309.57 nM T40492 CL9NS3 44399978 IC50 > 199526.23 nM T40492 C9YO4K 44399979 IC50 > 199526.23 nM T40492 CX8M3O 44400003 IC50 = 39810.72 nM T40492 C4X1OG 44400004 IC50 = 19952.62 nM T40492 C5EV1S 44400005 IC50 = 158489.32 nM T40492 CFRU27 44400006 IC50 = 199526.23 nM T40492 C7FO3T 44400007 IC50 = 251188.64 nM T40492 CA6P2U 44400008 IC50 = 100000 nM T40492 CQP47M 44400009 IC50 = 7943.28 nM T40492 CCRB97 44400010 IC50 = 3981.07 nM T40492 CT40SR 44400033 IC50 = 31622.78 nM T40492 CA96HO 44400076 IC50 > 1000000 nM T40492 CX7O2Z 44400112 IC50 > 199526.23 nM T40492 C6Z5NC 44400113 IC50 > 199526.23 nM T40492 C6PCE5 44400114 IC50 = 31622.78 nM T40492 C95CRD 44400115 IC50 = 19952.62 nM T40492 CW5G3Z 73347065 IC50 > 50000 nM T40492 C6TNQ8 135412361 IC50 = 800 nM T40492 C53AWL 135434400 IC50 = 100 nM T05031 D09XZB 123631 IC50 > 50000 nM T05031 D0B3HD 2519 IC50 = 400000 nM T05031 D0E3SH 6918837 IC50 > 10000 nM T05031 D0E6XR 3062316 IC50 > 50000 nM T05031 D0F8RA 2153 IC50 = 800000 nM T05031 D0J5VR 11625818 IC50 = 281 nM T05031 D0R0MW 5329102 IC50 > 50000 nM T05031 D0RU0O 50905713 IC50 = 85 nM T05031 D0S5LD 135565596 IC50 = 3.7 nM T05031 D0W5HK 216239 IC50 > 50000 nM T05031 D01PGR 16123056 IC50 = 113 nM T05031 D01QSO 16654980 IC50 = 166 nM T05031 D03BHZ 52913813 IC50 = 3 nM T05031 D03EZE 25167777 IC50 = 1.2 nM T05031 D03FOP 68947304 IC50 = 2700 nM T05031 D03KAC 1893730 IC50 = 383 nM T05031 D03LWG 53235510 IC50 > 9000 nM T05031 D03XAQ 49784945 IC50 = 120 nM T05031 D06GUA 49784002 IC50 = 1584.89 nM T05031 D07EHV 44814409 IC50 > 9100 nM T05031 D07HPJ 11476171 IC50 > 9000 nM T05031 D08QGT 17755052 IC50 = 33 nM T05031 D0C3ZR 10427712 IC50 = 1200 nM T05031 D0D8JB 44516953 IC50 = 6 nM T05031 D0E6UZ 54575456 IC50 = 16 nM T05031 D0G3MN 56949517 IC50 = 0.89 nM T05031 D0I3LO 91933883 IC50 = 82 nM T05031 D0O1LD 11647372 IC50 = 6 nM T05031 D0O6VZ 25254071 IC50 = 27 nM T05031 D0TU7B 58507717 IC50 = 661 nM T05031 D0U3DP 46912230 IC50 = 68 nM T05031 D0U3EP 445154 IC50 = 500 nM T05031 D0UP1Z 51001932 Ki = 9.1 nM T05031 D0VG0D 11977753 IC50 = 6 nM T05031 D0W7HE 56649450 IC50 = 1200 nM T05031 D0X7IN 11978790 IC50 = 63 nM T05031 D0XD4I 118502708 IC50 = 1800 nM T05031 D0Y2NS 70798655 IC50 = 4500 nM T05031 D03BNU 59604787 IC50 > 5000 nM T05031 D05HIJ 135565159 IC50 = 23 nM T05031 D09SFV 3973 IC50 = 270 nM T05031 D0D0QA 44137675 IC50 = 10 nM T05031 D0P1JI 312145 IC50 = 10 nM T05031 C3FRX9 131989 IC50 = 21000 nM T05031 C05RDN 566479 IC50 = 14200 nM T05031 CY3D4G 617191 IC50 = 3581 nM T05031 CS5O7B 622000 IC50 > 40000 nM T05031 CXC3V1 622262 IC50 = 693 nM T05031 C0S3EF 721057 IC50 = 130000 nM T05031 CU73NO 736009 IC50 = 81000 nM T05031 CIL9P1 913795 IC50 > 100000 nM T05031 C0L5VC 946390 IC50 = 3000 nM T05031 CWOQ49 1627922 IC50 = 10000 nM T05031 CKCW93 2612441 IC50 > 100000 nM T05031 C09VKD 2816900 IC50 = 30000 nM T05031 CK79GO 2988969 IC50 = 12000 nM T05031 C1O4KS 4416330 IC50 = 23000 nM T05031 CIN5F7 4904109 IC50 <= 10000 nM T05031 C1YJM9 4912089 IC50 = 32000 nM T05031 CE74CV 5059890 IC50 = 100000 nM T05031 C2OZ0W 6484194 IC50 = 17000 nM T05031 CK2IR4 6852165 IC50 = 11000 nM T05031 CE1Y8A 9815659 IC50 = 2800 nM T05031 CC4F8I 10021687 IC50 = 2300 nM T05031 CZM84H 10066542 IC50 = 420 nM T05031 C2W9ED 10269329 IC50 = 150 nM T05031 C7SFI1 10296883 IC50 > 10000 nM T05031 C32NQS 10357196 IC50 = 6201 nM T05031 C72LGO 10432948 IC50 = 51 nM T05031 CAZT53 10475366 IC50 = 240 nM T05031 C7Z9HW 10832781 IC50 = 1540 nM T05031 CL8YE3 11230964 IC50 = 50000 nM T05031 C8Y6IM 11234514 IC50 = 432 nM T05031 CK65NF 11418892 IC50 > 9100 nM T05031 CL3Z4O 11419728 Ki = 90 nM T05031 CYBD21 11428504 IC50 = 110 nM T05031 CHJ30L 11492951 IC50 > 20000 nM T05031 C0O4SQ 11522078 IC50 = 20000 nM T05031 C7HMO6 11526786 IC50 = 13 nM T05031 C38YWS 11541283 IC50 = 1.28 nM T05031 C1VA4C 11543481 IC50 = 100000 nM T05031 CN2MS6 11562853 IC50 = 1584.89 nM T05031 CMVQ43 11576772 IC50 = 11 nM T05031 CEHZ82 11599141 IC50 = 5011.87 nM T05031 C1ZPM5 11630874 IC50 = 20000 nM T05031 CY8C9P 11751126 IC50 = 2336 nM T05031 CAJV97 11955205 IC50 = 14.3 nM T05031 CBR6D5 11955693 IC50 = 289 nM T05031 CH7XM1 11955694 IC50 > 1000 nM T05031 C68SND 11955695 IC50 = 1093 nM T05031 C60DBM 11998444 IC50 = 14020 nM T05031 C5FTB0 11998445 IC50 = 1609 nM T05031 C68WMR 11998447 IC50 = 11460 nM T05031 CYL24B 11998448 IC50 = 4200 nM T05031 CNPI54 11998563 IC50 > 50000 nM T05031 C6AK0Y 11998564 IC50 > 50000 nM T05031 CMVA72 11998565 IC50 = 6943 nM T05031 CJ3YP8 11998685 IC50 = 20730 nM T05031 CV8PB5 11998690 IC50 = 511 nM T05031 CB9T1H 11998803 IC50 = 1157 nM T05031 C59SKD 11999032 IC50 = 1006 nM T05031 CT58GS 12171624 IC50 > 1000 nM T05031 CY7A0T 14638904 IC50 = 100000 nM T05031 CW5FD8 16081736 IC50 = 1279 nM T05031 CV9US5 16736978 IC50 > 30000 nM T05031 C72THB 16739368 IC50 = 3 nM T05031 CF6JS9 16757570 IC50 = 1100 nM T05031 CB19TH 16757576 IC50 = 120 nM T05031 C9BJ7Q 16757577 IC50 = 16 nM T05031 C9DM4T 16757578 IC50 = 170 nM T05031 C1NZC7 16757579 IC50 = 32 nM T05031 CY0S6G 17751063 IC50 = 215 nM T05031 C1SN9M 17756679 IC50 >= 100000 nM T05031 C7M2XJ 22036837 IC50 = 41 nM T05031 CH2BE0 22036876 IC50 = 72 nM T05031 CVDL81 22036885 IC50 = 3.5 nM T05031 C61ZGT 22135435 IC50 > 50118.72 nM T05031 CP05ZB 22346757 IC50 = 100000 nM T05031 C1F2TM 23582995 IC50 = 3360 nM T05031 CEYL29 23585510 Ki = 250 nM T05031 COW91A 23586721 IC50 = 4200 nM T05031 CBL37C 23642173 Ki = 340 nM T05031 C8J1SI 23642272 IC50 = 450 nM T05031 C59CTR 23652981 IC50 = 35 nM T05031 C29SFI 24768579 IC50 = 1919 nM T05031 CL4C8H 24809743 IC50 > 10000 nM T05031 CP4G9Z 24855584 Ki = 860 nM T05031 CM9C0R 24866805 IC50 = 50000 nM T05031 C8E9DQ 24880629 IC50 = 36000 nM T05031 CB79YC 24905143 IC50 = 8600 nM T05031 C2DC9J 24905144 IC50 = 16000 nM T05031 CN6V8Z 24905145 IC50 = 240 nM T05031 CSB7P5 24905148 IC50 = 15000 nM T05031 CGSF21 24905149 IC50 = 670 nM T05031 CVDG02 24905150 IC50 > 50000 nM T05031 CWH6C5 24905152 IC50 = 240 nM T05031 C0HE2Q 24905153 IC50 = 130 nM T05031 C7QSC9 24905154 IC50 = 5800 nM T05031 CO9D0K 24905155 IC50 = 3300 nM T05031 C5W9UR 24905157 IC50 = 80000 nM T05031 CA72BE 24905162 IC50 = 2100 nM T05031 CQN6X9 24905163 IC50 = 50000 nM T05031 CD4O1F 24905165 IC50 = 440 nM T05031 CKL48T 24905166 IC50 = 100000 nM T05031 C76VYL 24905167 IC50 = 7200 nM T05031 C7K5PU 24905168 IC50 = 1500 nM T05031 CZ57ID 24905169 IC50 = 100000 nM T05031 C2DHX9 24905170 IC50 = 50000 nM T05031 CSB96E 24905171 IC50 = 100000 nM T05031 CWZ0R2 24905172 IC50 = 1400 nM T05031 CY3B6M 24905175 IC50 = 3210 nM T05031 CW7UA3 24905176 IC50 = 1280 nM T05031 CW1V0H 24905177 IC50 = 100000 nM T05031 CO6Y0L 24905178 IC50 = 100000 nM T05031 C60NQW 24905179 IC50 = 1610 nM T05031 C4MO8B 24905180 IC50 = 5810 nM T05031 COJI47 24905181 IC50 = 5610 nM T05031 CS0B2C 24905182 IC50 = 343 nM T05031 C1H4BT 24905183 IC50 = 2880 nM T05031 C4WHK9 24905184 IC50 = 50300 nM T05031 C7Q4MZ 24905185 IC50 = 45000 nM T05031 CS4IP1 24905186 IC50 = 255 nM T05031 C69QWO 24905187 IC50 = 100000 nM T05031 C85ANB 24905188 IC50 = 3220 nM T05031 CNHD75 24905189 IC50 = 232 nM T05031 C9JUO2 24905190 IC50 = 4750 nM T05031 CPR03K 24905191 IC50 = 10600 nM T05031 CTAG19 24905193 IC50 = 4100 nM T05031 C7VJM5 24905194 IC50 = 46800 nM T05031 CEP1L3 24905195 IC50 = 67200 nM T05031 CP68ZD 24905196 IC50 = 28700 nM T05031 C8Z0RJ 24905197 IC50 = 3180 nM T05031 CN9RT0 24905198 IC50 = 100000 nM T05031 CHI78P 24905200 IC50 = 16000 nM T05031 CO6PE8 24905201 IC50 = 5000 nM T05031 CZ63HS 24905202 IC50 = 1000 nM T05031 C2X0FC 24905203 IC50 = 1000 nM T05031 C0WCE3 24905204 IC50 = 1400 nM T05031 CNK50B 24905205 IC50 = 2700 nM T05031 C12DPB 24905206 IC50 = 1900 nM T05031 C8N0RH 24905207 IC50 = 5300 nM T05031 CYA5G2 24905208 IC50 = 1600 nM T05031 CDV2B4 24905209 IC50 = 2900 nM T05031 CEFK68 24905210 IC50 = 1600 nM T05031 CUFP12 24905211 IC50 = 2700 nM T05031 C0JG8L 24905212 IC50 = 7000 nM T05031 CP47MK 24905213 IC50 = 100000 nM T05031 CB61QC 24905214 IC50 = 100000 nM T05031 CQ13ZI 24905215 IC50 = 100000 nM T05031 C6VI8F 24905216 IC50 = 5500 nM T05031 CXNH25 24905217 IC50 = 1300 nM T05031 C2PN9S 24905218 IC50 = 975 nM T05031 C9O2AL 24905219 IC50 = 476 nM T05031 CIT7U8 24905220 IC50 = 100000 nM T05031 CMD26S 24905221 IC50 = 854 nM T05031 C4R8WC 24905222 IC50 = 1100 nM T05031 C47SHA 24905223 IC50 = 550 nM T05031 C1DY2R 24905224 IC50 = 1500 nM T05031 CS0XF9 24905225 IC50 = 6500 nM T05031 CG5VX2 24905226 IC50 = 15000 nM T05031 C57QEO 24905227 IC50 = 100000 nM T05031 C7CG5E 24905228 IC50 = 4600 nM T05031 CHP5D1 24905229 IC50 = 25000 nM T05031 CXP09S 24905230 IC50 = 1100 nM T05031 CY7XG1 24905231 IC50 = 8900 nM T05031 C7JFQ2 24905232 IC50 = 500 nM T05031 C2JM1P 24905233 IC50 = 12000 nM T05031 CC3BF0 24905234 IC50 = 8100 nM T05031 CE57FI 24905235 IC50 = 7200 nM T05031 CUP20O 24905236 IC50 = 100000 nM T05031 CLC6Q2 24905237 IC50 = 100000 nM T05031 C9M1GI 24905238 IC50 = 5900 nM T05031 CVD72F 24905239 IC50 = 658 nM T05031 CK38IZ 24905240 IC50 = 742 nM T05031 CO2V5E 24905241 IC50 = 9200 nM T05031 CZBA19 24905244 IC50 = 548 nM T05031 CQ8OI1 24905246 IC50 = 52000 nM T05031 C5URC6 24905247 IC50 = 100000 nM T05031 C03SVO 24905250 IC50 = 50000 nM T05031 CIF2J5 24905251 IC50 = 3500 nM T05031 CPTE58 24905252 IC50 = 14200 nM T05031 CX1JB8 24905253 IC50 = 23000 nM T05031 COZ3H7 24905254 IC50 = 100000 nM T05031 CDT1H9 24905255 IC50 = 50000 nM T05031 C54QKA 24905256 IC50 = 25000 nM T05031 CRU3P2 24905257 IC50 = 100000 nM T05031 C9U0JA 24905259 IC50 = 100000 nM T05031 CO4YS7 24905260 IC50 = 100000 nM T05031 CEG0B5 24905261 IC50 = 100000 nM T05031 C9VE5F 24905262 IC50 = 100000 nM T05031 C3I4HK 24905264 IC50 = 100000 nM T05031 C0VMI6 24905265 IC50 = 100000 nM T05031 CWE3V0 24905267 IC50 = 100000 nM T05031 CH4T3A 24905268 IC50 = 100000 nM T05031 C6QDN7 24905271 IC50 = 50000 nM T05031 C6XHJ7 24905272 IC50 = 32000 nM T05031 CTB9A3 24905273 IC50 = 50000 nM T05031 C0NB1Q 24905274 IC50 = 50000 nM T05031 C9KQ0L 24905275 IC50 = 100000 nM T05031 C9O8QZ 24905277 IC50 = 30000 nM T05031 CP50RD 24905280 IC50 = 613 nM T05031 CG13ZM 24905281 IC50 = 5230 nM T05031 CF0S6X 24905282 IC50 = 1670 nM T05031 C5HBL0 24905284 IC50 = 100000 nM T05031 C2Z5DN 24905285 IC50 = 5870 nM T05031 CL6GH8 24905286 IC50 = 1360 nM T05031 CKYO98 24905287 IC50 = 1720 nM T05031 CRNQ65 24905288 IC50 = 697 nM T05031 COD7I5 24905289 IC50 = 5290 nM T05031 C4LP7E 24905290 IC50 = 3130 nM T05031 CE9JC2 24905291 IC50 = 216 nM T05031 C2GI1R 24905292 IC50 = 4820 nM T05031 CHW8C4 24905293 IC50 = 809 nM T05031 CQF0H1 24905294 IC50 = 261 nM T05031 CNO7X0 24905295 IC50 = 660 nM T05031 C5WRG7 24905296 IC50 = 294 nM T05031 CQ1S0U 24905297 IC50 = 2450 nM T05031 C4UES7 24905298 IC50 = 9860 nM T05031 CMS69P 24905299 IC50 = 100000 nM T05031 CC0U5M 24905300 IC50 = 941 nM T05031 CW7X6S 24905301 IC50 = 5690 nM T05031 C97IQV 24905302 IC50 = 1020 nM T05031 CSJ47V 24905303 IC50 = 2700 nM T05031 CPN74C 24905304 IC50 = 6980 nM T05031 C5CS3N 24905305 IC50 = 962 nM T05031 CK4XE9 24905307 IC50 = 2820 nM T05031 CTU6Z3 24905308 IC50 = 100000 nM T05031 C9SQX1 24905309 IC50 = 432 nM T05031 CM75JP 24905310 IC50 = 1420 nM T05031 C9Q2BJ 24905311 IC50 = 2270 nM T05031 C9VUA1 24905312 IC50 = 864 nM T05031 CU3RS1 24905313 IC50 = 2670 nM T05031 CYG3H2 24905314 IC50 = 364 nM T05031 CV5Q7O 24905315 IC50 = 1240 nM T05031 C8SA3O 24905316 IC50 = 949 nM T05031 CI5MN3 24905317 IC50 = 550 nM T05031 CJ1P7K 24905318 IC50 = 809 nM T05031 C1T6YQ 24905319 IC50 = 1860 nM T05031 CAU86X 24905320 IC50 = 715 nM T05031 C54ISY 24905321 IC50 = 6470 nM T05031 C2GE5I 24905322 IC50 = 3620 nM T05031 C8D6YK 24905323 IC50 = 16300 nM T05031 C5NZH9 24905324 IC50 = 3530 nM T05031 C9D6JR 24905325 IC50 = 1580 nM T05031 CLZT41 24905326 IC50 = 1350 nM T05031 CW8FD3 24905327 IC50 = 100000 nM T05031 CHB7A2 24905328 IC50 = 481 nM T05031 CA8EI3 24905329 IC50 = 169 nM T05031 CCQ0O7 24905330 IC50 = 525 nM T05031 CJ81AS 24905331 IC50 = 173 nM T05031 C8PW4H 24905332 IC50 = 235 nM T05031 C2Y5TF 24905333 IC50 = 320 nM T05031 CH9FL5 24905334 IC50 = 3800 nM T05031 C1S0PC 24905335 IC50 = 5400 nM T05031 C8N9MV 24905336 IC50 = 4600 nM T05031 C9E8BJ 24905338 IC50 = 5200 nM T05031 CX85AC 24905341 IC50 = 6100 nM T05031 CKZ80E 24905342 IC50 = 350 nM T05031 CO8SH1 24905343 IC50 = 230 nM T05031 C7IZL6 24905344 IC50 = 6100 nM T05031 C43VSW 24936353 IC50 = 501.19 nM T05031 C98MEW 24946175 IC50 = 27 nM T05031 CC7H3U 24946706 IC50 = 6.2 nM T05031 CDWQ10 24947414 Ki = 108 nM T05031 C78NJE 24955795 IC50 = 5344 nM T05031 C8P6NT 24956158 IC50 = 7991 nM T05031 CJI29P 24956159 IC50 = 5309 nM T05031 C8QPN6 24992904 IC50 = 194 nM T05031 C6C4RH 24993871 IC50 = 14 nM T05031 CEW91Q 25032963 IC50 = 23 nM T05031 CY50OT 25052783 IC50 = 540 nM T05031 CHR51O 25057242 IC50 = 1900 nM T05031 CD69RK 25097993 IC50 = 220 nM T05031 CV1N4E 25109782 Ki = 39 nM T05031 CLP07J 25110819 IC50 > 10000 nM T05031 CLS7P0 25129381 IC50 = 19952.62 nM T05031 C9R2EA 25129383 IC50 > 100000 nM T05031 C2CXH3 25165371 IC50 > 30000 nM T05031 CL87JW 25165773 IC50 > 30000 nM T05031 CB89TL 25165774 IC50 > 30000 nM T05031 CFZI92 25165961 IC50 > 30000 nM T05031 CK2YI4 25168990 IC50 = 5495.41 nM T05031 C7G1ZM 25169579 IC50 = 5450 nM T05031 CL81FJ 25169580 IC50 = 4420 nM T05031 C8WL0Z 25169784 IC50 > 1000 nM T05031 CLR8M2 25169786 IC50 > 1000 nM T05031 CL3UK2 25170000 IC50 > 1000 nM T05031 C6WCR7 25170003 IC50 = 44 nM T05031 C5PTZ0 25170410 IC50 > 1000 nM T05031 CLJR80 25171641 IC50 > 10000 nM T05031 C7ZQC2 25171642 IC50 > 1000 nM T05031 C7AHP4 25171644 IC50 > 1000 nM T05031 CX6BL8 25171852 IC50 > 1000 nM T05031 C7TL2N 25171853 IC50 > 1000 nM T05031 C6BR3F 25171855 IC50 = 390 nM T05031 CMI85O 25171856 IC50 = 230 nM T05031 CUN9F3 25171857 IC50 = 370 nM T05031 CKY81J 25172061 IC50 > 1000 nM T05031 CC1D8V 25172062 IC50 = 46 nM T05031 C1L6GX 25172063 IC50 = 1200 nM T05031 CFO08N 25172065 IC50 = 60 nM T05031 C8ZF0A 25172066 IC50 > 1000 nM T05031 CCW80B 25172270 IC50 > 1000 nM T05031 C9HUB6 25172271 IC50 = 550 nM T05031 CC60ZY 25172272 IC50 = 620 nM T05031 C54EGX 25172274 IC50 > 1000 nM T05031 C5QVC7 25172275 IC50 = 830 nM T05031 CPW2D9 25172477 IC50 = 51 nM T05031 CVDC60 25172479 IC50 = 620 nM T05031 CI6W9H 25172661 IC50 = 62 nM T05031 CL5IC0 25172662 IC50 > 1000 nM T05031 CDAO95 25172663 IC50 = 490 nM T05031 C8JC3P 25172664 IC50 = 68 nM T05031 CK38ER 25172665 IC50 = 67 nM T05031 C3JI1Y 25172666 IC50 = 79 nM T05031 CLW96O 25207689 IC50 = 86 nM T05031 CWP29U 25242324 IC50 = 12 nM T05031 CARX27 25253230 IC50 = 332 nM T05031 C96OGS 25260915 IC50 = 141 nM T05031 CUR93V 25261554 IC50 = 2629 nM T05031 C3IDN0 25266674 IC50 = 15848.93 nM T05031 C2IM0O 39733146 IC50 = 15848.93 nM T05031 CIF63E 42623219 IC50 = 2511.89 nM T05031 C3DNM9 42623223 IC50 = 199.53 nM T05031 CG8Q0C 42630822 IC50 = 8100 nM T05031 C10RBA 42636535 IC50 = 6500 nM T05031 C3ROX1 44124863 Ki = 3.5 nM T05031 CI3K7H 44129042 IC50 > 9100 nM T05031 CIE0J3 44129043 IC50 > 9100 nM T05031 CUW85V 44129044 IC50 = 7100 nM T05031 C2B9DE 44129118 IC50 = 8000 nM T05031 C6O0JA 44129197 IC50 = 5000 nM T05031 C0R1PH 44129198 IC50 > 9100 nM T05031 C6LGD5 44129200 IC50 = 8600 nM T05031 C03RLS 44129270 IC50 > 9100 nM T05031 CTG8U7 44129271 IC50 = 4900 nM T05031 CDQ56T 44129272 IC50 > 9100 nM T05031 CU4H1I 44129274 IC50 > 9100 nM T05031 C79QOC 44129275 IC50 = 7000 nM T05031 C0W3ZF 44129348 IC50 > 9100 nM T05031 CQ5UJ4 44129350 IC50 = 2100 nM T05031 CH6RO4 44129351 IC50 > 9100 nM T05031 CPAU59 44129353 IC50 > 9100 nM T05031 CN5O4I 44129429 IC50 = 5500 nM T05031 CON25C 44129430 IC50 = 8900 nM T05031 C3ZSV2 44129432 IC50 = 8500 nM T05031 C3MWZ1 44129511 IC50 > 9100 nM T05031 CM5U2I 44137407 IC50 = 693 nM T05031 CF17OS 44180029 IC50 = 632 nM T05031 CHK8Z6 44180034 IC50 = 1750 nM T05031 CEJ5F7 44180035 IC50 = 568 nM T05031 CQNT23 44180155 IC50 = 7047 nM T05031 CIKM57 44180156 IC50 = 214 nM T05031 CBP2T3 44180157 IC50 = 371 nM T05031 C2S5LC 44180395 IC50 = 195 nM T05031 C40NOQ 44180397 IC50 = 433 nM T05031 CTB46H 44180398 IC50 = 3600 nM T05031 CE30IL 44180626 IC50 = 244 nM T05031 CRS2G3 44180853 IC50 = 1161 nM T05031 C9HU7V 44181276 IC50 = 240 nM T05031 C2VZX7 44181492 IC50 = 150 nM T05031 C7SYM2 44181493 IC50 = 1027 nM T05031 CB8KF1 44181494 IC50 = 2554 nM T05031 C5AI8R 44181598 IC50 = 134 nM T05031 CK03RW 44181599 IC50 > 50000 nM T05031 CXL61J 44181600 IC50 = 378 nM T05031 C6TZK5 44181601 IC50 = 367 nM T05031 CCIV74 44181602 IC50 = 310 nM T05031 C36WUP 44181603 IC50 = 9247 nM T05031 CL6W0C 44181605 IC50 = 2757 nM T05031 CFD41Z 44181718 IC50 = 5241 nM T05031 C2RB1P 44181719 IC50 = 1205 nM T05031 CMC75I 44181720 IC50 > 50000 nM T05031 CWTS93 44181721 IC50 = 175 nM T05031 CT1JL2 44181722 IC50 = 418 nM T05031 CE9HO1 44181723 IC50 = 139 nM T05031 CFSB29 44181724 IC50 = 161 nM T05031 C96DJK 44241762 Ki = 643 nM T05031 C92UIQ 44241764 Ki = 2900 nM T05031 CFC1E3 44242168 Ki = 144 nM T05031 CJ27VR 44242423 Ki = 582 nM T05031 CT6AD8 44242428 Ki = 114 nM T05031 CM1Z7F 44242776 Ki = 199 nM T05031 CJ8QI0 44242777 Ki = 31 nM T05031 C98MAL 44436951 IC50 > 10000 nM T05031 CD0ME6 44436952 IC50 > 10000 nM T05031 CR6ZU9 44436953 IC50 > 10000 nM T05031 CYK0T1 44436954 IC50 > 10000 nM T05031 CYV15O 44436955 IC50 > 10000 nM T05031 C3M4RN 44436961 IC50 > 10000 nM T05031 CA4SV2 44436964 IC50 > 10000 nM T05031 CO5FK1 44436967 IC50 > 10000 nM T05031 CRKU98 44436970 IC50 > 10000 nM T05031 C9V1SZ 44436971 IC50 > 10000 nM T05031 CZ4V2L 44436972 IC50 > 10000 nM T05031 COG34Q 44436976 IC50 > 10000 nM T05031 C4RAK8 44436979 IC50 > 10000 nM T05031 CXN93Q 44436980 IC50 > 10000 nM T05031 CX57RI 44436981 IC50 > 10000 nM T05031 C9ZML1 44454396 IC50 = 446 nM T05031 C30NZA 44475985 IC50 = 316 nM T05031 CAT8F7 44475986 IC50 = 23 nM T05031 CSR73H 44475987 IC50 = 750 nM T05031 CDAX92 44475988 IC50 = 664 nM T05031 CBH0S5 44475989 IC50 = 4230 nM T05031 CW5A7L 44475990 IC50 = 9 nM T05031 C03IGD 44540030 IC50 = 31622.78 nM T05031 C5LWU1 44540126 IC50 = 19952.62 nM T05031 CYD4Z8 44540130 IC50 = 1000 nM T05031 CAT2R7 44540316 IC50 = 12589.25 nM T05031 C2T9GC 44540407 IC50 = 6309.57 nM T05031 CQ4PE7 44540492 IC50 = 25118.86 nM T05031 CH3L9P 44551660 IC50 = 5440 nM T05031 C3VRO9 44557921 IC50 = 489.78 nM T05031 CRE61W 44577592 IC50 = 2001 nM T05031 CH63GM 44577593 IC50 = 376 nM T05031 CA8MV5 44577594 IC50 = 1625 nM T05031 C9IXW8 44577638 IC50 = 1048 nM T05031 C8A5RT 44577639 IC50 = 452 nM T05031 CNP02V 44577640 IC50 = 308 nM T05031 CT6GN5 44577641 IC50 = 623 nM T05031 CIQR97 44577850 IC50 = 1226 nM T05031 CCG8P9 44577851 IC50 = 11690 nM T05031 CLBA40 44577853 IC50 = 1245 nM T05031 COU6V7 44577854 IC50 = 1621 nM T05031 C8M5FY 44577914 IC50 = 1448 nM T05031 CGO09K 44577916 IC50 = 3656 nM T05031 CRJ3B7 44577917 IC50 = 834 nM T05031 CTR89C 44577918 IC50 = 10320 nM T05031 CO05YG 44577919 IC50 = 727 nM T05031 CT70WA 44577920 IC50 = 298 nM T05031 C5KXS4 44577921 IC50 = 1470 nM T05031 CZ2HI5 44577922 IC50 = 325 nM T05031 CGTU34 44577950 IC50 = 3521 nM T05031 CQC50R 44577951 IC50 = 336 nM T05031 C8ZTW2 44577952 IC50 = 1593 nM T05031 CIL93G 44577953 IC50 = 964 nM T05031 C8NB5H 44578037 IC50 > 40000 nM T05031 CX9TO2 44578038 IC50 = 4163 nM T05031 C7AHR4 44578039 IC50 > 50000 nM T05031 C13LGI 44578040 IC50 > 50000 nM T05031 CNZ06H 44578074 IC50 > 50000 nM T05031 C41TYA 44578108 IC50 = 481 nM T05031 C2W3SQ 44578109 IC50 = 2545 nM T05031 C40VHS 44580686 IC50 = 222 nM T05031 C0L2HO 44593630 IC50 = 1325 nM T05031 C2NQ6Z 44593631 IC50 = 156 nM T05031 CY3SV7 44596118 IC50 > 30000 nM T05031 CH6V9F 44608754 IC50 = 15 nM T05031 C0IY9N 44608757 IC50 = 9.8 nM T05031 C90ITS 44608915 IC50 = 13 nM T05031 CZH1P9 44609387 IC50 = 15 nM T05031 CNDX48 44609388 IC50 = 9.6 nM T05031 C2ISK4 44610761 IC50 > 100000 nM T05031 CE95RQ 44620964 IC50 = 14 nM T05031 CVYJ36 44620965 IC50 = 60 nM T05031 CA8BY7 44621440 IC50 = 31622776.6 nM T05031 C5M1FR 44621441 IC50 = 63095734.45 nM T05031 C5LD7E 44621442 IC50 = 25118864.32 nM T05031 CO4GT0 44621447 IC50 = 39810717.06 nM T05031 CUV26H 44621448 IC50 = 12589254.12 nM T05031 CV2MG9 44621449 IC50 = 31622776.6 nM T05031 C24IYW 44621451 IC50 = 31622776.6 nM T05031 C0F9YW 44621452 IC50 = 25118864.32 nM T05031 C0GRD8 44621454 IC50 = 39810717.06 nM T05031 C4YHJ0 44621456 IC50 = 39810717.06 nM T05031 C31VBF 44621458 IC50 = 31622776.6 nM T05031 CP6DB9 45265864 IC50 = 850 nM T05031 CZ68MG 45488079 IC50 > 10000 nM T05031 CV1U7I 46180604 IC50 = 38 nM T05031 CED2B3 46180606 IC50 = 5400 nM T05031 CDV85O 46180663 IC50 = 1400 nM T05031 CZGB46 46180666 IC50 = 25 nM T05031 CAU17V 46202808 IC50 = 1258.93 nM T05031 CDA3R9 46220225 IC50 = 31 nM T05031 C7RF5Y 46239967 IC50 > 1000 nM T05031 C94YRI 46853654 IC50 = 398.11 nM T05031 CZ3WS1 46861592 IC50 = 0.2 nM T05031 C63RCG 46870269 IC50 = 1000 nM T05031 CTQ25M 46871497 IC50 = 1258.93 nM T05031 CQB16A 46872415 IC50 > 20000 nM T05031 C3HMQ2 46891474 IC50 = 0.7 nM T05031 CB6Z8P 46892208 IC50 = 15400 nM T05031 CZX46Y 46892342 IC50 = 1400 nM T05031 C5FN6I 46892845 IC50 = 870 nM T05031 CQ32BN 46892970 IC50 = 9 nM T05031 COJA32 46892971 Ki = 43 nM T05031 C5QFB3 46893088 IC50 = 630 nM T05031 CS30AI 46893754 IC50 = 8500 nM T05031 CJ0VB4 46932297 IC50 = 4400 nM T05031 CF14PE 46947264 IC50 = 24 nM T05031 COE37N 49778924 EC50 = 6.31 nM T05031 C7ZK3D 49783923 IC50 = 630.96 nM T05031 CHX76J 49784892 Ki = 23 nM T05031 CA1H8S 49784893 Ki = 51 nM T05031 CP2QD0 49784894 Ki = 5 nM T05031 CTZG05 49784988 Ki = 9 nM T05031 CE9AC5 49785078 Ki = 130 nM T05031 CG2IO7 49785079 Ki = 28 nM T05031 C8EYN4 49785083 Ki = 7 nM T05031 CZI34V 49785167 Ki = 990 nM T05031 CJK65T 49785253 Ki = 35 nM T05031 CXK8F5 49785436 Ki = 3 nM T05031 CWL5C6 49785518 Ki = 6 nM T05031 C3NV0J 49785827 Ki = 3 nM T05031 C0OZM2 49785828 Ki = 17 nM T05031 C1AR4G 49785829 Ki = 2300 nM T05031 C90JBE 49834576 IC50 = 547 nM T05031 C9ZW3R 49835055 IC50 = 1130 nM T05031 C5UR4A 49843944 IC50 = 140 nM T05031 CS40YB 49853846 IC50 = 1000 nM T05031 C7PER0 49853953 IC50 = 1400 nM T05031 CU9A8O 49854022 IC50 = 262 nM T05031 C51QVH 49854023 IC50 = 20 nM T05031 CM4HQ2 49854024 IC50 = 387 nM T05031 C1LBX3 49854049 IC50 = 75 nM T05031 CVC2H6 49854052 IC50 = 220 nM T05031 CC2X9N 49854121 IC50 = 469 nM T05031 CAJ58E 49854156 IC50 = 730 nM T05031 CAU39Y 49854158 IC50 = 280 nM T05031 CPK6X3 49854360 IC50 = 2500 nM T05031 CBVT70 49854361 IC50 = 720 nM T05031 CQ1TZ6 49854365 IC50 = 1300 nM T05031 CJ5I9X 49854461 IC50 = 450 nM T05031 CDXQ69 49854462 IC50 = 4500 nM T05031 C0ORZ9 49854466 IC50 = 2300 nM T05031 CY14XF 49854572 IC50 = 770 nM T05031 CEC10T 49854573 IC50 = 220 nM T05031 C39KQW 49854679 IC50 = 670 nM T05031 C8VDR2 49854680 IC50 = 930 nM T05031 CN2V8R 49854681 IC50 = 5500 nM T05031 CSN96A 49855001 IC50 = 2000 nM T05031 CALY90 49855192 IC50 > 9100 nM T05031 CJPE20 49855193 IC50 = 4600 nM T05031 C1OM3I 49855237 IC50 = 540 nM T05031 CY8MP7 49867926 IC50 = 113 nM T05031 CR0IA5 49871864 IC50 > 20000 nM T05031 C13WJZ 49872243 IC50 = 710 nM T05031 C5OY7B 49872246 IC50 = 545 nM T05031 C2KD5E 49872344 IC50 = 280 nM T05031 CV5BF3 49872645 IC50 = 1240 nM T05031 CN97FO 49872646 IC50 = 1100 nM T05031 CD6P5R 49872735 IC50 = 2720 nM T05031 CL64NB 49872737 IC50 = 17000 nM T05031 CRNG04 49872831 IC50 = 8.2 nM T05031 CQC8B4 49872835 IC50 = 420 nM T05031 CPS3O1 49872924 IC50 = 460 nM T05031 CUBX74 49872925 IC50 = 500 nM T05031 CAW69U 49872927 IC50 = 510 nM T05031 CV1L4P 49873242 IC50 = 7160 nM T05031 C5BA2V 49873243 IC50 = 4610 nM T05031 CSN45W 49873329 IC50 = 143 nM T05031 C9CW7X 50908894 IC50 = 240 nM T05031 CLC2N7 50913517 IC50 = 2340 nM T05031 CJ4L8Y 50938829 Ki > 125000 nM T05031 CJG65L 50939078 IC50 = 36 nM T05031 CI8QM1 50939080 IC50 = 10 nM T05031 CT0IP3 50939081 Ki = 54 nM T05031 C8JD5T 50939209 IC50 = 39 nM T05031 C54EUL 50939212 Ki = 395 nM T05031 CS7Z6U 50939338 Ki = 30 nM T05031 CXT23Y 50939344 IC50 = 105 nM T05031 C6GH4K 50939865 IC50 = 59 nM T05031 C2I9PS 50939992 IC50 = 60 nM T05031 C9TUE4 50940108 IC50 = 81 nM T05031 CQ93GK 50940110 IC50 = 35 nM T05031 CG4R5C 50940334 IC50 = 60 nM T05031 C2Q0GE 50990922 Ki = 190 nM T05031 CKY3V1 50990924 Ki = 2 nM T05031 C5ZF9W 51003380 IC50 = 4800 nM T05031 CY36EH 51003592 IC50 = 1584.89 nM T05031 CLB85F 51346892 IC50 = 1600 nM T05031 C65ILG 51346893 IC50 = 100 nM T05031 C9MO5I 51601993 IC50 = 6 nM T05031 CA1PL9 51601994 IC50 = 800 nM T05031 CT91WR 52040626 IC50 > 1000 nM T05031 CD84MT 52913592 IC50 = 49 nM T05031 C2TLG6 52913931 IC50 = 12 nM T05031 CU1P2L 52940797 IC50 = 100000 nM T05031 C2KI6V 52942202 IC50 = 100000 nM T05031 CDHJ08 52942235 IC50 = 7000 nM T05031 C4VCY0 52943258 IC50 = 100000 nM T05031 C1XEV2 52943394 IC50 = 2640 nM T05031 CHI0P6 52944356 IC50 = 100000 nM T05031 C4NLX7 52945630 IC50 = 492 nM T05031 CXD6T8 52945845 IC50 = 8000 nM T05031 C7ET6Z 52948010 IC50 = 15000 nM T05031 CV5B2C 52949497 IC50 = 25000 nM T05031 CH1Q5D 53234281 IC50 = 5.5 nM T05031 C45JKN 53234283 IC50 = 20.3 nM T05031 CVK28S 53235062 IC50 = 7.9 nM T05031 COW61E 53235216 IC50 = 32.4 nM T05031 CWE56X 53235217 IC50 = 13 nM T05031 CDXM59 53235451 IC50 = 63 nM T05031 CT8IN1 53242225 IC50 = 4500 nM T05031 C4J9WZ 53307606 Ki = 19 nM T05031 CRD3A9 53316967 IC50 = 440 nM T05031 C84YNK 53317325 IC50 = 17000 nM T05031 CS8DJ3 53318252 IC50 = 200 nM T05031 C7JB1A 53318613 IC50 = 48000 nM T05031 C58NQJ 53318614 IC50 = 62000 nM T05031 C10YUH 53318615 IC50 = 9000 nM T05031 CFJD70 53319932 IC50 = 17000 nM T05031 C3EJB1 53319933 IC50 = 12000 nM T05031 C2V7AX 53320017 IC50 = 5200 nM T05031 CKGJ60 53320018 IC50 = 370 nM T05031 CJRM64 53322563 IC50 = 17000 nM T05031 CN92LK 53322732 IC50 = 92 nM T05031 CY6L1D 53323901 IC50 = 57000 nM T05031 CJZ29M 53325374 IC50 = 2600 nM T05031 C1TE8J 53325515 IC50 = 2300 nM T05031 C6LAI9 53326166 IC50 = 1900 nM T05031 C23HAU 53361718 IC50 = 10 nM T05031 CM60WQ 53361719 IC50 = 15 nM T05031 C6Q8RC 53378051 IC50 = 794.33 nM T05031 CVG90B 53389651 IC50 > 10000 nM T05031 CSV9X2 54579940 IC50 = 17 nM T05031 CN51TL 54579941 IC50 = 28800 nM T05031 C7VZU2 54579942 IC50 = 3100 nM T05031 C4R9JB 54579943 IC50 = 1000 nM T05031 CG26HQ 54579944 IC50 = 3700 nM T05031 CC5R3O 54580924 IC50 = 1000 nM T05031 C3OIY4 54580925 IC50 = 1000 nM T05031 C60TYL 54581049 IC50 = 1000 nM T05031 CF2UH5 54581983 IC50 = 410 nM T05031 C23EVN 54582916 IC50 = 1800 nM T05031 CT2SV7 54583916 IC50 = 1030 nM T05031 CY87EC 54583917 IC50 = 2400 nM T05031 C8CPI4 54584859 IC50 = 22300 nM T05031 C9TZ2V 54584860 IC50 = 6900 nM T05031 CME81Q 54585830 IC50 = 420 nM T05031 CQE3L1 54669876 Ki = 204 nM T05031 CE4TS9 56589559 IC50 = 1.4 nM T05031 C8JK0C 56593675 IC50 = 94 nM T05031 CW3SK6 56593676 IC50 = 118 nM T05031 C45WYD 56593677 IC50 = 0.91 nM T05031 CW65IM 56593678 IC50 = 18.5 nM T05031 C8UQH2 56593830 IC50 = 170 nM T05031 CV5FQ7 56593831 IC50 = 40 nM T05031 COJ1V2 56595026 IC50 = 1030 nM T05031 CE2NY1 56595155 IC50 = 53 nM T05031 CN0H7L 56595156 IC50 = 461 nM T05031 CE4GU0 56595157 IC50 = 39 nM T05031 CW6R7J 56595158 IC50 = 230 nM T05031 CW5J7M 56595159 IC50 = 250 nM T05031 CZG5B4 56595160 IC50 > 1000 nM T05031 C89JUC 56595290 IC50 = 383 nM T05031 C3Z5GJ 56595293 IC50 = 104 nM T05031 C3D4OZ 56595294 IC50 = 518 nM T05031 CM5P4R 56595420 IC50 = 2400 nM T05031 CR24WQ 56595421 IC50 = 56 nM T05031 CE4HG2 56595422 IC50 = 2100 nM T05031 C4XZ1B 56595423 IC50 = 570 nM T05031 CWJK79 56595424 IC50 = 480 nM T05031 C4YAJ0 56595547 IC50 > 1000 nM T05031 CMIK83 56595548 IC50 = 68 nM T05031 CL9K0Z 56595549 IC50 = 310 nM T05031 C6IOX2 56595550 IC50 > 1000 nM T05031 C3R9PW 56595551 IC50 > 1000 nM T05031 C1OSZ8 56595682 IC50 > 1000 nM T05031 C2KWD4 56595683 IC50 > 1000 nM T05031 CND5I4 56595684 IC50 = 47 nM T05031 C3G5RZ 56595685 IC50 = 801 nM T05031 CJ41GT 56595686 IC50 = 6.7 nM T05031 C2PN4S 56599298 IC50 = 4150 nM T05031 CT64SR 56599306 IC50 = 36 nM T05031 CFUT05 56648675 IC50 = 11 nM T05031 C1GAB6 56648677 IC50 = 29 nM T05031 CWDF40 56648757 IC50 = 44 nM T05031 CE35CB 56648758 IC50 = 19 nM T05031 CJO39U 56648759 IC50 = 45 nM T05031 CNKC90 56654649 IC50 = 1330 nM T05031 CE2Q5Y 56673546 Ki = 87 nM T05031 CQME43 56680186 Ki = 272 nM T05031 C94JIT 56832510 IC50 = 8.6 nM T05031 CC9IP6 56833458 Ki = 69 nM T05031 CKD9T4 56833539 Ki = 1167 nM T05031 CLG1W9 56833540 Ki = 41 nM T05031 C7GMY3 56833541 Ki = 7 nM T05031 CI0LP9 56833542 Ki = 18 nM T05031 CE2XW4 56833543 Ki = 25 nM T05031 C6PK0Z 56833544 Ki = 42 nM T05031 C07XMA 56833636 Ki = 43 nM T05031 C7RA0U 56833637 Ki = 247 nM T05031 CBHQ53 56833638 Ki = 55 nM T05031 CY7Q6N 56833639 Ki = 33 nM T05031 CPDO94 56833738 Ki = 30 nM T05031 C5C6QT 56833739 Ki = 55 nM T05031 CK36WM 56833740 Ki = 3870 nM T05031 C0IJP8 56927258 EC50 = 1000 nM T05031 C9MJG4 56929824 IC50 = 7 nM T05031 CYFB96 56932203 IC50 = 2511.89 nM T05031 C8C2FG 56932238 IC50 = 19952.62 nM T05031 CX6Q2K 56932240 IC50 = 251.19 nM T05031 CO6K5Q 56955953 IC50 > 10000 nM T05031 CAK91L 56955954 IC50 = 2059 nM T05031 C8B6JG 56955955 IC50 > 10000 nM T05031 CW8B4D 57330208 IC50 = 2800 nM T05031 C6JMN9 57345685 IC50 = 2 nM T05031 CZ7RE0 57345686 IC50 = 1 nM T05031 CA53SC 57351276 Ki = 1410 nM T05031 C1X3UP 57390135 IC50 > 1000 nM T05031 CQ6N8D 57390136 IC50 = 480 nM T05031 C6XDC8 57390137 IC50 > 1000 nM T05031 C0S6IG 57390138 IC50 = 230 nM T05031 C2RI4V 57390139 IC50 > 1000 nM T05031 CZ3FU2 57390175 IC50 > 1000 nM T05031 CR2X7O 57390176 IC50 > 1000 nM T05031 CK2SO6 57390300 IC50 = 0.81 nM T05031 C1GVK3 57391362 IC50 = 250 nM T05031 CLHX38 57391363 IC50 = 80 nM T05031 C0PR9J 57391364 IC50 = 32 nM T05031 C6L9HO 57391365 IC50 = 90 nM T05031 C2QX0T 57391366 IC50 = 1000 nM T05031 CLQ9J1 57391367 IC50 = 6 nM T05031 C53HZJ 57391915 IC50 > 1000 nM T05031 CO18UJ 57391916 IC50 = 410 nM T05031 CRU8Q0 57391917 IC50 = 600 nM T05031 C13DRO 57391952 IC50 > 1000 nM T05031 CH8UV4 57391962 IC50 = 280 nM T05031 CB2KF3 57392078 IC50 = 35 nM T05031 CQ1W0C 57393124 IC50 = 4 nM T05031 CZ0RW2 57393125 IC50 = 2000 nM T05031 C3G9VK 57393643 IC50 > 1000 nM T05031 CJX56V 57393644 IC50 = 30 nM T05031 CAND02 57393679 IC50 > 1000 nM T05031 CA93ZE 57394864 IC50 = 25 nM T05031 CF6C2T 57395364 IC50 > 1000 nM T05031 CKE35B 57395365 IC50 > 1000 nM T05031 CWL2D6 57395366 IC50 > 1000 nM T05031 CB6L7N 57395397 IC50 > 1000 nM T05031 CJH9S2 57395408 IC50 > 1000 nM T05031 C31MCE 57395409 IC50 = 300 nM T05031 CSP45C 57395410 IC50 = 44 nM T05031 CDG2F3 57396625 IC50 = 3 nM T05031 CD73TE 57396626 IC50 = 100 nM T05031 CQRU75 57396627 IC50 = 40 nM T05031 CI34XH 57396628 IC50 = 13 nM T05031 C92FYK 57397192 IC50 > 1000 nM T05031 CBC7N6 57397236 IC50 > 1000 nM T05031 CK01SI 57397253 IC50 = 64 nM T05031 C3Q2ZP 57398390 IC50 = 400 nM T05031 C56TEZ 57398391 IC50 = 40 nM T05031 CP9Q4U 57398392 IC50 = 63 nM T05031 C0O5KE 57398393 IC50 = 100 nM T05031 C5PI3B 57398894 IC50 > 1000 nM T05031 COTK97 57398895 IC50 > 1000 nM T05031 CD5Z7P 57399042 IC50 = 25 nM T05031 C3G9HW 57399126 IC50 = 79 nM T05031 CYE09F 57400062 IC50 = 6 nM T05031 CN5PY7 57400063 IC50 = 32 nM T05031 CT0Y7E 57400064 IC50 = 20 nM T05031 C0PZM5 57400579 IC50 > 1000 nM T05031 C9BW8C 57400580 IC50 = 340 nM T05031 C4K2RZ 57400581 IC50 > 1000 nM T05031 C4MW8J 57400582 IC50 > 1000 nM T05031 CGC91E 57400641 IC50 = 63 nM T05031 CM63CS 57401865 IC50 = 13 nM T05031 CG6M4H 57401867 IC50 = 100 nM T05031 CP8FY5 57401868 IC50 = 2 nM T05031 CQ5P4X 57401869 IC50 = 13 nM T05031 C2X8PO 57402386 IC50 = 1800 nM T05031 CNMV98 57402387 IC50 = 130 nM T05031 C06IYP 57402428 IC50 = 360 nM T05031 CF68RN 57403576 IC50 = 400 nM T05031 CL2R7T 57403577 IC50 = 25 nM T05031 CC5N9R 57403578 IC50 = 8 nM T05031 CZ8M5F 57403579 IC50 = 32 nM T05031 C5NT7R 57403580 IC50 = 25 nM T05031 CHBV63 57403581 IC50 = 1 nM T05031 CAC72X 57403582 IC50 = 320 nM T05031 CNR95F 57404840 IC50 > 9100 nM T05031 CED47A 57410062 IC50 = 11 nM T05031 C1BVX6 57411134 IC50 = 25 nM T05031 C39JSW 57411135 IC50 = 45 nM T05031 CL8F6Q 57411137 IC50 = 40 nM T05031 CW97FT 57411139 IC50 = 38 nM T05031 CU0R3A 57411250 IC50 = 1420 nM T05031 C6C5TU 57411252 IC50 = 340 nM T05031 CD0W2I 57411254 IC50 = 11 nM T05031 CW1DA3 57411255 IC50 = 110 nM T05031 C6U4LO 57411256 IC50 = 22 nM T05031 CP9G7L 57411366 IC50 = 75 nM T05031 CC5DO3 57411369 IC50 = 2000 nM T05031 C56RBS 57411372 IC50 = 49 nM T05031 CX9O3T 57411485 IC50 = 308 nM T05031 CQBM65 57411486 IC50 = 240 nM T05031 CK5QX7 57411488 IC50 = 25 nM T05031 C90LNK 57411715 IC50 = 15 nM T05031 CPXE40 57411716 IC50 = 876 nM T05031 CE6RY5 57411836 IC50 = 14 nM T05031 C5JOX3 57411837 IC50 = 10 nM T05031 C0I5JM 57419280 IC50 > 10000 nM T05031 CT6XL0 57466811 Ki = 320 nM T05031 CRB5P2 57495287 IC50 = 1710 nM T05031 C59YAC 57495353 IC50 = 424 nM T05031 CMT9L7 57495355 IC50 = 951 nM T05031 CWQ6F2 57523291 IC50 = 1333 nM T05031 CJE19S 57523686 IC50 = 739 nM T05031 C6L4FZ 57599744 IC50 = 4000 nM T05031 CV9J7D 57748162 IC50 = 1200 nM T05031 CL57CP 57789333 IC50 = 2300 nM T05031 C81BYH 57798309 IC50 = 1100 nM T05031 CZ21KP 57900314 IC50 = 29 nM T05031 C8S7NQ 58203695 IC50 = 3.9 nM T05031 CO20YT 58203712 IC50 = 9.3 nM T05031 CINT74 58203776 IC50 = 9.2 nM T05031 C7X0OJ 58203779 IC50 = 8.4 nM T05031 C36IVB 58203785 IC50 = 14 nM T05031 C61ZNP 58203789 IC50 = 13 nM T05031 CF85YJ 58203795 IC50 = 7.4 nM T05031 CEM32T 58203808 IC50 = 8.5 nM T05031 C5KLV8 58203898 IC50 = 1.8 nM T05031 CG65RS 58203922 IC50 = 4 nM T05031 CW1M9X 58203976 IC50 = 5.4 nM T05031 COFN62 58203995 IC50 = 17.4 nM T05031 CN8D9F 58204007 IC50 = 7 nM T05031 CPDQ83 58204017 IC50 = 2.4 nM T05031 C16GRS 58204034 IC50 = 37.8 nM T05031 CM62NB 58204076 IC50 = 0.9 nM T05031 C07NXV 58204082 IC50 = 7.6 nM T05031 C81XIQ 58204138 IC50 = 1.8 nM T05031 C8Y4RB 58204237 IC50 = 4.6 nM T05031 CGA01N 58204242 IC50 = 3.9 nM T05031 C4MK5I 58204259 IC50 = 14.2 nM T05031 CVR9Q2 58233988 IC50 = 251.19 nM T05031 CB9AH8 58234990 IC50 = 19 nM T05031 CJ8YI2 58234995 IC50 = 11 nM T05031 CZF3U5 58235016 IC50 = 12 nM T05031 CM0ND7 58235018 IC50 = 7 nM T05031 C25RXY 58235020 IC50 = 15 nM T05031 CAY94U 58235030 IC50 = 13 nM T05031 CAJC03 58235033 IC50 = 9 nM T05031 CN7MZ8 58235039 IC50 = 11 nM T05031 CPW84H 58235041 IC50 = 10 nM T05031 C70CRN 58235043 IC50 = 100 nM T05031 C5SQV3 58235052 IC50 = 10 nM T05031 CEZ4T5 58235053 IC50 = 33 nM T05031 C82LIS 58235061 IC50 = 9 nM T05031 C3SO4E 58235062 IC50 = 15 nM T05031 CZ0SD5 58235073 IC50 = 10 nM T05031 CQP25T 58235077 IC50 = 2 nM T05031 C0LDZ2 58235079 IC50 = 128 nM T05031 C2YG5L 58235088 IC50 = 12 nM T05031 CJ6R8Q 59251679 IC50 = 270 nM T05031 CRZ5B1 59251991 IC50 = 2940 nM T05031 CILJ94 59293648 IC50 = 1920 nM T05031 C6A3KL 59293676 IC50 = 3100 nM T05031 CC14ZL 59293709 IC50 = 4100 nM T05031 C0R3TX 59293715 IC50 = 4000 nM T05031 C9TVC6 59293721 IC50 = 5500 nM T05031 CZ5OV1 59293740 IC50 = 4400 nM T05031 CB2Z4R 59293755 IC50 = 3900 nM T05031 C8AL6C 59293763 IC50 = 1800 nM T05031 CT3CF1 59477024 IC50 = 19952.62 nM T05031 C7KG5E 59477042 IC50 = 25118.86 nM T05031 C2X8TY 59548177 Ki = 11 nM T05031 CGRO45 59548196 Ki = 65 nM T05031 CD39AG 59548207 Ki = 9700 nM T05031 C6KP4G 59548220 Ki = 41 nM T05031 CTNU85 59548226 Ki = 86 nM T05031 CLB6N4 59548232 Ki > 10000 nM T05031 CSWV07 59548243 Ki = 44 nM T05031 CMT2R0 59548250 Ki = 320 nM T05031 C3I8NE 59548256 Ki = 59 nM T05031 C8W5HT 59548263 Ki = 580 nM T05031 CT8Q5B 59548274 Ki = 89 nM T05031 CVF1B2 59548283 Ki = 81 nM T05031 CY31EA 59548284 Ki = 67 nM T05031 CO4GT7 59548288 Ki = 0.6 nM T05031 CFR7S8 59548302 Ki = 56 nM T05031 CRM20Z 59548320 Ki = 22 nM T05031 CJE5I4 59548341 Ki = 75 nM T05031 C8O1VS 59548349 Ki = 5 nM T05031 CWC65A 59548356 Ki = 5 nM T05031 CMKP95 59548371 Ki = 15 nM T05031 CC8UV3 59548383 Ki = 45 nM T05031 CD4ET2 59548402 Ki = 130 nM T05031 CES59T 59548403 Ki = 740 nM T05031 CE8P3G 59548407 Ki = 16 nM T05031 CO4K2W 59548419 Ki = 4.7 nM T05031 CSDB78 59548424 Ki = 15 nM T05031 C81FCQ 59548431 Ki = 7 nM T05031 CLGY34 59548453 Ki = 48 nM T05031 CBT21W 59548454 Ki = 110 nM T05031 CJT68K 59548460 Ki = 38 nM T05031 C9LFT3 59548462 Ki = 2 nM T05031 CX8C2U 59548480 Ki = 1300 nM T05031 C4Y3GL 59609976 IC50 = 8930 nM T05031 C1PC0J 59634638 IC50 > 20000 nM T05031 CP2UY3 59634686 IC50 = 2840 nM T05031 C1TH2N 59634692 IC50 = 240 nM T05031 CPA0L2 59634709 IC50 = 11000 nM T05031 CBI0M6 59688563 IC50 = 1584.89 nM T05031 COFZ83 59753763 IC50 = 210 nM T05031 CUYB59 60148924 IC50 > 10000 nM T05031 CM8PD7 60150509 IC50 = 0.3 nM T05031 C5KD3Z 60154714 Ki > 10000 nM T05031 CS0L4D 60154996 Ki > 10000 nM T05031 C1UI3P 60155086 Ki > 10000 nM T05031 CX08ON 60155087 Ki = 610 nM T05031 CX8J1I 60155265 Ki = 20 nM T05031 CAT40I 60155266 Ki = 9 nM T05031 CD56VA 60155268 Ki = 7 nM T05031 CCQB56 60155375 IC50 = 1970 nM T05031 CH5X2S 60155376 IC50 = 3512 nM T05031 C74FEN 60155377 IC50 = 2970 nM T05031 CZ6G4B 60155378 IC50 = 578 nM T05031 C10AHQ 60155379 IC50 = 1563 nM T05031 C5FI4P 60155451 Ki = 18 nM T05031 CX9G4U 60155452 Ki = 16 nM T05031 C9Q7DE 60155469 IC50 = 701 nM T05031 CH8UY5 60155470 IC50 = 2511 nM T05031 C3EDY4 60155471 IC50 > 10000 nM T05031 CE0ZX1 60155472 IC50 = 3370 nM T05031 CG90MC 60155473 IC50 = 362 nM T05031 C82PVI 60155474 IC50 > 10000 nM T05031 CX49FT 60155475 IC50 = 6343 nM T05031 CR7EG9 60155538 Ki = 61 nM T05031 CU6YB9 60155539 Ki = 13 nM T05031 CW6N1S 60155552 IC50 = 64 nM T05031 CIB08V 60155553 IC50 = 2075 nM T05031 CZE28G 60155554 IC50 = 1611 nM T05031 CZD2W7 60155555 IC50 = 1656 nM T05031 CO6IU3 60155556 IC50 = 5070 nM T05031 C6HN5O 60155557 IC50 = 1130 nM T05031 CMQ9G1 60155638 IC50 = 2404 nM T05031 CG56KT 60155639 IC50 = 1263 nM T05031 CBJ65P 60155640 IC50 = 4774 nM T05031 C8OJK0 60155641 IC50 = 1069 nM T05031 CT9XJ6 60155642 IC50 = 4442 nM T05031 C5BYQ3 60155643 IC50 = 1964 nM T05031 C57RBF 60155722 IC50 = 1968 nM T05031 CU7J6L 60155723 IC50 = 5016 nM T05031 CSZA16 60155724 IC50 = 1148 nM T05031 C21DWT 60155725 IC50 = 6275 nM T05031 C12CQU 60155726 IC50 = 2643 nM T05031 CA5TM3 60155805 IC50 = 54 nM T05031 C60RIO 60155806 IC50 = 39 nM T05031 CIRO73 66493714 IC50 = 603 nM T05031 C71LPV 66493729 IC50 = 946 nM T05031 CRC24S 66552467 IC50 = 199526.23 nM T05031 C46POH 66552523 IC50 > 100000 nM T05031 C68LXT 66552524 IC50 > 100000 nM T05031 C91JZL 66553214 IC50 = 42 nM T05031 CUC7B3 66557964 IC50 = 1.1 nM T05031 C6YPT5 66558054 IC50 = 1.2 nM T05031 C9X2TB 66558056 IC50 = 2.8 nM T05031 CD64VW 66559243 IC50 = 1.2 nM T05031 C1R3SI 66653673 IC50 = 9870 nM T05031 CF8BZ7 66677439 IC50 = 300 nM T05031 CN0RE8 66779813 IC50 = 0.5 nM T05031 C3IP5D 66779815 IC50 = 0.5 nM T05031 CH86MR 66779905 IC50 = 3 nM T05031 CX2N6E 66779920 IC50 = 79 nM T05031 C9O4TC 66779989 EC50 = 6 nM T05031 CF2UM8 66780001 IC50 = 50 nM T05031 CHU0C5 66780007 EC50 = 3 nM T05031 CGL4V1 66780016 IC50 = 3 nM T05031 C5F6OA 66780027 IC50 = 320 nM T05031 C8DN7A 66780034 IC50 = 790 nM T05031 C4AM6R 66780100 EC50 = 16 nM T05031 CZ5P2N 66780118 IC50 = 0.05 nM T05031 CREA54 66780266 IC50 = 10 nM T05031 CRCA72 66780292 IC50 = 0.3 nM T05031 CW2SM6 66780337 EC50 = 6 nM T05031 CU54DY 66780379 IC50 = 3 nM T05031 CQ70YA 66780434 IC50 = 3 nM T05031 C8F9UY 66780515 IC50 = 0.2 nM T05031 CFH6C2 66780644 IC50 = 25 nM T05031 CTZB46 66780835 IC50 = 160 nM T05031 CEP5A2 66780844 IC50 = 8 nM T05031 C51ARE 66788835 Ki = 17 nM T05031 CS4Q3G 66839776 IC50 = 9 nM T05031 CE9N0C 66839794 IC50 = 190 nM T05031 C9SUG0 66839801 IC50 = 17 nM T05031 CUJ5Z4 66839834 IC50 = 81 nM T05031 CW12XO 66882257 IC50 = 104 nM T05031 C6IO1S 66883557 IC50 = 244 nM T05031 C1HSE0 67035086 IC50 = 230 nM T05031 C38RGB 67035556 IC50 > 9000 nM T05031 CV3HW2 67035568 IC50 > 9000 nM T05031 C8HOZ9 67041250 IC50 > 30000 nM T05031 C5E4AJ 67050504 IC50 = 77 nM T05031 CMWO25 67061712 IC50 = 15 nM T05031 C0OX5N 67103709 IC50 = 6 nM T05031 C9J2EO 67103712 IC50 = 1 nM T05031 CM4W1Y 67103722 IC50 = 7 nM T05031 C5TYQ3 67103909 IC50 = 0.4 nM T05031 CVJ49E 67103974 IC50 = 10 nM T05031 C3VFY7 67104025 IC50 = 7 nM T05031 CC07KA 67104052 IC50 = 12 nM T05031 C7EZW6 67192973 IC50 = 7 nM T05031 C1OXI2 67284515 IC50 = 143 nM T05031 CQHF85 67284779 IC50 = 53 nM T05031 C3K4DG 67285093 IC50 = 720 nM T05031 CYD3P9 67285103 IC50 = 54 nM T05031 CT6BX3 67285457 Ki = 269 nM T05031 C25AHY 67984037 IC50 > 9100 nM T05031 C8I7GC 68293638 IC50 > 10000 nM T05031 CI1HJ5 68504925 IC50 > 1000 nM T05031 C01QHM 68547896 IC50 = 130 nM T05031 CAR46Z 70675172 IC50 = 295 nM T05031 C0L9EF 70675845 IC50 = 2600 nM T05031 CN09DI 70675846 IC50 = 38 nM T05031 C6BQE1 70681248 IC50 = 1.3 nM T05031 CPE36T 70681262 IC50 = 1 nM T05031 CPX41V 70682086 IC50 = 125.89 nM T05031 CQW54O 70682591 Ki = 1360 nM T05031 CPV59G 70682592 Ki > 10000 nM T05031 CB3ZN5 70683337 IC50 = 2.5 nM T05031 C1I5PH 70683338 IC50 = 2 nM T05031 CSM0A6 70684204 IC50 = 63.1 nM T05031 CXD08N 70684690 Ki = 870 nM T05031 C8O2QH 70685440 IC50 = 1.3 nM T05031 CZG9M1 70685441 IC50 = 13 nM T05031 CH7KO0 70685442 IC50 = 0.4 nM T05031 C6G4WB 70686339 IC50 > 100000 nM T05031 CON8X4 70686340 IC50 = 3162.28 nM T05031 C1ASW4 70686341 IC50 = 79.43 nM T05031 C0PWL5 70686455 IC50 > 1000 nM T05031 CN4CR2 70686584 IC50 = 3 nM T05031 C85FWA 70686829 Ki = 410 nM T05031 CQS8G7 70686830 Ki = 2000 nM T05031 CH62EI 70687595 IC50 = 2 nM T05031 C8QSD2 70688455 IC50 > 199.53 nM T05031 CFCJ02 70688558 IC50 > 199.53 nM T05031 CSX6I7 70688908 Ki = 1430 nM T05031 C5YN6U 70689166 IC50 = 400 nM T05031 C6L4WY 70689639 IC50 = 0.6 nM T05031 CGT1X2 70690496 IC50 = 630.96 nM T05031 CW3U5J 70690994 Ki = 1940 nM T05031 CC6I1Q 70691259 IC50 = 790 nM T05031 CD3JL4 70691776 IC50 = 1.6 nM T05031 CDK52M 70692650 IC50 > 1995.26 nM T05031 C3TM1F 70693128 Ki = 1300 nM T05031 C2VAU8 70693129 Ki = 550 nM T05031 C65FHO 70694723 Ki = 94.1 nM T05031 CPFO83 70694805 IC50 = 398.11 nM T05031 CRNY76 70695188 Ki = 760 nM T05031 C3N5YJ 70695189 Ki > 10000 nM T05031 C75YGN 70695469 IC50 = 5 nM T05031 C61CFG 70696737 IC50 = 1000 nM T05031 C7KL5X 70696852 IC50 = 3981.07 nM T05031 CRH8E2 71270723 EC50 = 158.49 nM T05031 CWR58A 71270783 IC50 = 39.81 nM T05031 CF9LU4 71270807 EC50 = 63.1 nM T05031 C7FDL2 71270817 IC50 = 2.512 nM T05031 CNR1G9 71270824 EC50 = 10000 nM T05031 C38LBA 71270831 IC50 = 0.3981 nM T05031 CTL6R5 71270836 EC50 = 19952.62 nM T05031 CM4LX7 71270848 EC50 = 1258.93 nM T05031 C2GWX6 71270906 IC50 = 794.33 nM T05031 CX0DL3 71270910 IC50 = 7.943 nM T05031 C0COW6 71270913 IC50 = 25.12 nM T05031 CB0S8G 71270927 IC50 = 0.3981 nM T05031 C24IOW 71270948 IC50 = 63.1 nM T05031 C5BJ2Y 71270957 IC50 > 1258.93 nM T05031 C03NFY 71271625 IC50 = 1000 nM T05031 CL47JU 71271739 IC50 = 12.59 nM T05031 CS5JG6 71271910 IC50 = 6.31 nM T05031 C4PSK8 71271965 IC50 = 2.512 nM T05031 CB4N1M 71272066 IC50 > 1258.93 nM T05031 CD8E1Y 71272453 EC50 = 1000 nM T05031 C8EW9V 71272757 IC50 = 316.23 nM T05031 C0LO8I 71272765 IC50 = 2.512 nM T05031 C42PJQ 71449564 IC50 = 29000 nM T05031 CFN52U 71449565 IC50 = 1500 nM T05031 C7ULC4 71449776 IC50 = 100 nM T05031 CNHJ63 71451228 IC50 > 10000 nM T05031 CLZO91 71451372 IC50 = 10000 nM T05031 CSB2E6 71451587 IC50 = 90 nM T05031 C9O5HM 71451588 IC50 = 3100 nM T05031 C19XDJ 71453176 IC50 = 25000 nM T05031 C71JEC 71453177 IC50 = 32000 nM T05031 CR84JX 71453419 Ki = 4 nM T05031 CEKG39 71453424 IC50 = 980 nM T05031 CF1B5X 71453425 IC50 = 1400 nM T05031 CZ61FJ 71454160 IC50 = 50118723.36 nM T05031 CZ8Q5P 71454238 Ki = 4.4 nM T05031 C4NS8G 71454916 IC50 = 34000 nM T05031 CIK32W 71454917 IC50 = 87000 nM T05031 CC46RH 71455124 IC50 = 140 nM T05031 CCP3M4 71455125 IC50 = 1200 nM T05031 C1ILO7 71456697 IC50 = 2500 nM T05031 C9ENV7 71456698 IC50 = 23000 nM T05031 CCPV51 71458543 IC50 = 110000 nM T05031 CMZA06 71458544 IC50 = 1600 nM T05031 CF42GC 71458545 IC50 = 36000 nM T05031 CD50NR 71458791 IC50 = 1000 nM T05031 C8ELG4 71460604 IC50 = 130 nM T05031 CS7VI3 71460605 IC50 = 970 nM T05031 CA7QI2 71460606 IC50 = 200 nM T05031 C1O2ET 71460607 IC50 = 220 nM T05031 CVQ26M 71462083 IC50 = 43000 nM T05031 CXLQ15 71462308 IC50 = 600 nM T05031 CU3EO6 71520393 IC50 = 214 nM T05031 CYC6S1 71520394 IC50 > 10000 nM T05031 C1KMX0 71520395 IC50 = 1790 nM T05031 CYK7N8 71520396 IC50 > 10000 nM T05031 CTC0O8 71520397 IC50 = 726 nM T05031 C0UZ3D 71526877 IC50 = 1000 nM T05031 CP05SQ 71526878 IC50 = 2800 nM T05031 CZK6X9 71526879 IC50 > 10000 nM T05031 C8QRE4 71526880 IC50 = 140 nM T05031 CT3QI8 71526881 IC50 = 220 nM T05031 CO4MY1 71527005 IC50 = 26 nM T05031 CJC64F 71527006 IC50 = 50 nM T05031 C96WZG 71527007 IC50 = 98 nM T05031 CUC7I1 71527008 IC50 = 260 nM T05031 C09WKC 71527009 IC50 = 2400 nM T05031 CSPO76 71527716 IC50 = 316.23 nM T05031 CIN7O1 71527842 IC50 > 3162.28 nM T05031 CO6CI7 71528725 IC50 = 35 nM T05031 C5U2ZC 71528726 IC50 = 54 nM T05031 CTKO36 71528727 IC50 = 62 nM T05031 CI7Q4K 71548718 IC50 = 3570 nM T05031 CED62L 71548719 IC50 = 1910 nM T05031 C4JPR6 71583220 IC50 = 1.585 nM T05031 C3X2PU 71610694 IC50 = 5.012 nM T05031 C4NGT1 71612553 IC50 = 435.86 nM T05031 C6PRV1 71655831 IC50 = 77 nM T05031 CWG8M3 71682651 IC50 = 1800 nM T05031 C6UGW3 71682652 IC50 > 9100 nM T05031 C7BX4K 71682653 IC50 = 4900 nM T05031 CQX8N3 71682654 IC50 = 8200 nM T05031 CCG6J1 71682807 IC50 > 9100 nM T05031 CS32HB 71716798 IC50 = 39.81 nM T05031 C07GCV 71716799 IC50 = 1258.93 nM T05031 CFW01E 71718034 IC50 = 419 nM T05031 C29KOU 72709209 IC50 > 10000 nM T05031 CT73IW 72709284 IC50 = 4500 nM T05031 C9P1IG 72943510 IC50 = 7052 nM T05031 C8EI1X 73673707 IC50 = 1.8 nM T05031 CBYN18 73977439 IC50 > 30000 nM T05031 C9V1YR 73977449 IC50 = 31623 nM T05031 CXA90D 73977451 IC50 = 7943 nM T05031 CEZ7L2 73977461 IC50 = 7943 nM T05031 CD0T9V 74539799 IC50 = 1.7 nM T05031 C16KOS 74539862 IC50 = 1.1 nM T05031 CIBQ59 76311315 IC50 > 1000 nM T05031 C8BD3K 76311316 IC50 = 140 nM T05031 C6F1CR 76311317 IC50 > 1000 nM T05031 C7IDU0 76311318 IC50 > 1000 nM T05031 CG40TB 76311319 IC50 > 1000 nM T05031 C5WSZ8 76311320 IC50 > 1000 nM T05031 C0M5SE 76311321 IC50 > 1000 nM T05031 CA2VR6 76311340 IC50 = 729 nM T05031 CCY5L6 76314906 IC50 > 1000 nM T05031 CE3Z1I 76314907 IC50 > 1000 nM T05031 CFY10G 76314908 IC50 > 1000 nM T05031 C4UHR5 76314909 IC50 = 4340 nM T05031 C1B3VO 76314910 IC50 > 1000 nM T05031 CY0Z4U 76314911 IC50 > 1000 nM T05031 CTVO82 76314912 IC50 > 1000 nM T05031 CCWP56 76314913 IC50 > 1000 nM T05031 CO13XZ 76314937 IC50 = 938 nM T05031 C7W2HI 76314938 IC50 > 1000 nM T05031 C6H9EL 76314939 IC50 = 673 nM T05031 C3SIE7 76318525 IC50 > 1000 nM T05031 CU6G7L 76318526 IC50 > 1000 nM T05031 CC3Z2U 76318527 IC50 = 3560 nM T05031 CS6ME5 76318566 IC50 = 839 nM T05031 CG4I2R 76318567 IC50 = 741 nM T05031 CR61ZP 76322185 IC50 > 1000 nM T05031 C5LT0B 76322186 IC50 > 1000 nM T05031 C19SKA 76322187 IC50 > 1000 nM T05031 C1YFK9 76322218 IC50 = 799 nM T05031 CL0T7B 76322219 IC50 = 373 nM T05031 C1HFI9 76325446 IC50 = 17 nM T05031 C7IFD5 76325803 IC50 > 1000 nM T05031 C2NK4S 76325804 IC50 > 1000 nM T05031 COJ6P9 76325805 IC50 > 1000 nM T05031 C2AJ6T 76325806 IC50 > 1000 nM T05031 C4GZ1Q 76325833 IC50 = 977 nM T05031 CQ31CA 76325834 IC50 = 874 nM T05031 C8S2IL 76329389 IC50 > 1000 nM T05031 CAEW42 76329390 IC50 > 1000 nM T05031 CMC32D 76329391 IC50 > 1000 nM T05031 CAZ9Q2 76329392 IC50 > 1000 nM T05031 C06ZQJ 76329393 IC50 > 1000 nM T05031 C39CLE 76329428 IC50 = 863 nM T05031 CE6BI0 76332666 IC50 = 307 nM T05031 CKG1E0 76333034 IC50 > 1000 nM T05031 C6D4RU 76333035 IC50 > 1000 nM T05031 CSAT72 76333036 IC50 > 1000 nM T05031 C1JRO2 76333037 IC50 > 1000 nM T05031 C8TNI0 76333038 IC50 > 1000 nM T05031 C16SRX 76333068 IC50 = 537 nM T05031 CW81MC 76333069 IC50 = 961 nM T05031 C26CKL 76333070 IC50 = 573 nM T05031 C47NLT 76333071 IC50 = 926 nM T05031 CP2UC5 76336660 IC50 > 1000 nM T05031 C79JAI 76336661 IC50 > 1000 nM T05031 CJ3V6Y 76336695 IC50 = 851 nM T05031 CD03GB 76336696 IC50 = 893 nM T05031 C2JTH8 77107528 IC50 = 589 nM T05031 C42HDP 77107927 IC50 = 241 nM T05031 C04SRC 77147259 IC50 = 736 nM T05031 C9I7TY 78319187 IC50 > 125892.54 nM T05031 C5P3RO 86647783 IC50 = 1800 nM T05031 CG3KJ4 86672407 IC50 = 2 nM T05031 C2QG3S 86672408 IC50 = 3 nM T05031 C8EA6S 86672420 IC50 = 2.3 nM T05031 C5K4RT 86672424 IC50 = 4.5 nM T05031 CDXM47 86677874 IC50 > 20000 nM T05031 CP3W1B 86695297 IC50 > 20000 nM T05031 CA17UE 86732669 IC50 = 1650 nM T05031 CV6PI8 87562294 IC50 = 251.19 nM T05031 C5L3ZP 89051724 IC50 = 3.2 nM T05031 C1HB3F 89051931 IC50 = 3.4 nM T05031 CTE1L0 89517065 IC50 = 380 nM T05031 C56KSC 89517226 IC50 = 6180 nM T05031 C08UWK 90665816 IC50 = 130 nM T05031 CMWB58 91757958 IC50 <= 10000 nM T05031 C3Y0DS 91801158 IC50 = 149 nM T05031 CAS7W6 91864650 IC50 > 20000 nM T05031 C67VQE 118341819 IC50 > 10000 nM T05031 CC9P5H 118341835 IC50 > 10000 nM T05031 CUMA23 118341844 IC50 = 670 nM T05031 C3IP9X 118341852 IC50 > 10000 nM T05031 C6TI0Z 118341865 IC50 > 10000 nM T05031 C4U7NC 118341870 IC50 > 10000 nM T05031 CVL03K 118341884 IC50 > 10000 nM T05031 CPZN96 118341923 IC50 > 10000 nM T05031 C9E3DU 118341927 IC50 > 10000 nM T05031 CCPV26 118575517 EC50 = 3.7 nM T05031 CEDC48 118575654 EC50 = 42 nM T05031 COYJ84 118575663 EC50 = 3.4 nM T05031 CUJ30I 118575784 EC50 = 4.2 nM T05031 CAT54V 118575791 EC50 = 15 nM T05031 CAD39P 118575986 EC50 = 7.6 nM T05031 CCYI54 118576050 EC50 = 45 nM T05031 CCJ91U 118709071 IC50 = 4800 nM T05031 CL4U2W 118709072 IC50 = 31 nM T05031 C2CE4Q 118709073 IC50 = 84 nM T05031 C05EHL 118709074 IC50 = 30 nM T05031 CVS6W4 118709075 IC50 = 12 nM T05031 CZ5SO8 118709076 IC50 = 59 nM T05031 CRX24W 118709077 IC50 = 11 nM T05031 C9IUX6 118709078 IC50 = 58 nM T05031 C7R9FA 118709079 IC50 = 140 nM T05031 CY14MF 118709080 IC50 = 340 nM T05031 CV2EJ7 118709081 IC50 = 8 nM T05031 C9RF7I 118709082 IC50 = 76 nM T05031 CVI98J 118709083 IC50 = 190 nM T05031 CLEB72 118709084 IC50 = 110 nM T05031 CV94YO 118709085 IC50 = 180 nM T05031 CO3F4B 118709086 IC50 = 660 nM T05031 CH4N9Y 118709087 IC50 = 1700 nM T05031 C8JZ7E 118709088 IC50 = 400 nM T05031 C52YKH 118709089 IC50 = 47 nM T05031 C94IZR 118709090 IC50 = 200 nM T05031 C0UTL3 118709091 IC50 = 46 nM T05031 CR6ML1 118709578 IC50 = 7 nM T05031 C0OH7I 118709579 IC50 = 37 nM T05031 CV3G7J 118709580 IC50 = 39 nM T05031 C7AG0Q 118709581 IC50 = 73 nM T05031 C73YIO 118709582 IC50 = 7 nM T05031 CGWX02 118709583 IC50 = 5 nM T05031 CZ87IH 118709584 IC50 = 11 nM T05031 CCAH61 118709585 IC50 = 11 nM T05031 CQ13GC 118709586 IC50 = 25 nM T05031 CXP2O5 118709587 IC50 = 8 nM T05031 CPN46D 118709588 IC50 = 25 nM T05031 CY64OB 118709589 IC50 = 29 nM T05031 C8N0TA 118709711 IC50 = 75 nM T05031 C9S7KX 118709712 IC50 = 10 nM T05031 CW91QF 118709713 IC50 = 7 nM T05031 CAN4K9 118709714 IC50 = 12 nM T05031 CP3WA1 118709715 IC50 = 2 nM T05031 CQ69PZ 118709716 IC50 = 23 nM T05031 C7LZV8 118709717 IC50 = 74 nM T05031 C3C0KF 118709718 IC50 = 530 nM T05031 CB53EU 118728320 IC50 = 907 nM T05031 C6KJL1 118728321 IC50 = 488 nM T05031 CKJ3S6 118728322 IC50 = 473 nM T05031 CT0L3Y 118728325 IC50 = 363 nM T05031 CHS2E4 118728326 IC50 = 188 nM T05031 CRUP47 118728328 IC50 = 1032 nM T05031 CQR41G 118728330 IC50 = 284 nM T05031 CN4Q9R 118728332 IC50 = 184 nM T05031 CDI10F 118728336 IC50 = 1213 nM T05031 CHT6K9 118728811 Ki > 4000 nM T05031 CUA3Y2 118728812 Ki > 4000 nM T05031 CDQ78G 118728813 Ki > 4000 nM T05031 CZ6XL7 118728814 Ki = 2000 nM T05031 CMO67K 118728815 Ki > 4000 nM T05031 CR2M0Q 118728816 Ki > 4000 nM T05031 C62SCL 118728817 Ki > 4000 nM T05031 CSB30C 118728819 Ki > 4000 nM T05031 CV7XU8 118728820 Ki = 2500 nM T05031 C3J1EX 118728821 Ki > 4000 nM T05031 CIWB78 118728822 Ki > 4000 nM T05031 CP18SE 118728823 Ki > 4000 nM T05031 CM42CA 118728824 Ki = 2300 nM T05031 C9Q7CL 118728825 Ki > 4000 nM T05031 CCR3S0 118728826 Ki > 4000 nM T05031 CB1WC5 118729946 IC50 = 160 nM T05031 CQ4G9M 118729947 IC50 = 5000 nM T05031 C43IPJ 118729948 IC50 = 230 nM T05031 C3I9CQ 118729949 IC50 = 280 nM T05031 CZQ17M 118729950 IC50 = 80 nM T05031 C3G1ZP 118729951 IC50 = 4030 nM T05031 CY60FC 118730033 IC50 = 394 nM T05031 CN3B4U 118730711 IC50 = 5 nM T05031 C0IL3N 118730712 IC50 = 13 nM T05031 C3CH1A 118730713 IC50 = 2 nM T05031 CHX5L9 118730714 IC50 = 3 nM T05031 CNJ32C 118730715 IC50 = 35 nM T05031 C1MKB3 118730716 IC50 = 7 nM T05031 C81RJA 118730717 IC50 = 17 nM T05031 CFZ16R 118737301 IC50 <= 10000 nM T05031 C27CPQ 118737302 IC50 <= 10000 nM T05031 C59VXA 118737303 IC50 <= 10000 nM T05031 CGO1N4 118737304 IC50 <= 10000 nM T05031 CS85FM 118737305 IC50 <= 10000 nM T05031 C8UCO1 118737306 IC50 <= 10000 nM T05031 CR0BZ2 118737307 IC50 <= 10000 nM T05031 C3N4DJ 118737308 IC50 <= 10000 nM T05031 CGY5B1 118737309 IC50 <= 10000 nM T05031 CG9Q1H 121320416 IC50 = 40600 nM T05031 C5MB7C 121426227 IC50 = 17 nM T05031 CR75XB 121426239 IC50 = 33 nM T05031 CDTK36 121426321 IC50 = 17 nM T05031 CA3EL7 121426350 IC50 > 513 nM T05031 CXZT09 121426376 IC50 = 316 nM T05031 C0HXU2 121426388 IC50 = 501 nM T05031 CFN12W 121445751 IC50 = 17 nM T05031 C04NDW 121445810 IC50 = 85.6 nM T05031 C81IFQ 122163152 IC50 > 100000 nM T05031 C2VGD5 122178120 IC50 = 22.5 nM T05031 C24XUZ 122178124 IC50 = 3.6 nM T05031 CN5AB3 122179486 IC50 = 700 nM T05031 CLEK13 122179487 IC50 = 398 nM T05031 C0OW8H 122179490 IC50 = 765 nM T05031 C0VD5F 122179491 IC50 = 125.9 nM T05031 CQ87FB 122179492 IC50 = 501 nM T05031 CBJ29X 122179493 IC50 > 10000 nM T05031 CA5N1B 122179494 IC50 = 790 nM T05031 CSTE64 122179689 IC50 = 20 nM T05031 CE2FM7 122179690 IC50 = 30 nM T05031 CZJ31R 122179691 IC50 = 30 nM T05031 CBOU30 122179692 IC50 = 20 nM T05031 CKWC74 122179693 IC50 = 240 nM T05031 C4CX7Z 122179694 IC50 = 4600 nM T05031 C48LYC 122179695 IC50 = 310 nM T05031 C3D5QM 122179696 IC50 = 2100 nM T05031 CW3DM7 122179697 IC50 = 7400 nM T05031 C6I3PB 122179698 IC50 = 4800 nM T05031 CCU6A4 122179699 IC50 = 570 nM T05031 C7WMC3 122179700 IC50 = 230 nM T05031 C86NOQ 122179701 IC50 = 1000 nM T05031 CAHY19 122179702 IC50 = 1400 nM T05031 C3O7CM 122179703 IC50 = 1000 nM T05031 CK2R4X 122179704 IC50 = 450 nM T05031 CG96HD 122179705 IC50 = 670 nM T05031 C1PK9L 122179706 IC50 = 1200 nM T05031 CEB69W 122179707 IC50 = 3200 nM T05031 CK97EL 122179708 IC50 = 2100 nM T05031 C0ZA4C 122179709 IC50 = 1800 nM T05031 CU93YJ 122179710 IC50 = 590 nM T05031 C0KTH8 122179711 IC50 = 3600 nM T05031 CN9I1C 122179712 IC50 = 1500 nM T05031 C65OGI 122179713 IC50 = 3900 nM T05031 C92AZK 122179714 IC50 > 10000 nM T05031 CWL43Z 122179715 IC50 > 10000 nM T05031 C50VNH 122179716 IC50 > 10000 nM T05031 COW37C 122179717 IC50 > 10000 nM T05031 CG5N9E 122179718 IC50 = 1800 nM T05031 CB14FW 122179719 IC50 = 2400 nM T05031 CHZ3S1 122179720 IC50 = 1800 nM T05031 CEG8Y6 122179721 IC50 = 1900 nM T05031 CG5P3J 122179722 IC50 > 10000 nM T05031 CZH3T1 122179723 IC50 = 630 nM T05031 C10FGR 122179724 IC50 = 9100 nM T05031 CEFS13 122180793 IC50 = 26180 nM T05031 CFZ2E1 122180794 IC50 = 58430 nM T05031 C5YKG7 122180795 IC50 = 113450 nM T05031 C9ID7U 122180796 IC50 = 78290 nM T05031 C08XOC 122180839 IC50 = 323450 nM T05031 C2HM6P 122180840 IC50 = 418160 nM T05031 CT9Y6U 122180841 IC50 = 890 nM T05031 C6FOM0 122180842 IC50 = 560 nM T05031 COX90L 122180843 IC50 = 340 nM T05031 CP40RU 122180844 IC50 = 780 nM T05031 CC0EK9 122180845 IC50 = 480 nM T05031 CS85CU 122181413 IC50 = 900 nM T05031 CJ4T5W 122181414 IC50 = 10000 nM T05031 CK8L4D 122181415 IC50 = 650 nM T05031 CQS67B 122181416 IC50 = 6900 nM T05031 CB2AG9 122181417 IC50 = 12000 nM T05031 CFET49 122181418 IC50 = 1300 nM T05031 CQU14E 122181419 IC50 = 380 nM T05031 C58XRY 122184465 IC50 = 6309.57 nM T05031 C16ALM 122184466 IC50 = 5011.87 nM T05031 CIX19J 122184467 IC50 = 15848.93 nM T05031 CDZY02 122184468 IC50 = 79432.82 nM T05031 CTH70U 122184469 IC50 = 31622.78 nM T05031 C9ZXR7 122184470 IC50 = 12589.25 nM T05031 CNJ9Z4 122184471 IC50 = 39810.72 nM T05031 CS41EG 122184473 IC50 = 2511.89 nM T05031 CZ36GL 122184474 IC50 = 3981.07 nM T05031 CU4ZT6 122184475 IC50 = 39810.72 nM T05031 C3H9PR 122184476 IC50 = 6309.57 nM T05031 CU40TW 122184477 IC50 = 7943.28 nM T05031 CAMD31 122184479 IC50 = 79432.82 nM T05031 C1F9RK 122184480 IC50 = 1258.93 nM T05031 CQ7W0P 122184526 IC50 = 6309.57 nM T05031 CA5YB2 122184529 IC50 = 15848.93 nM T05031 C64YPH 122184530 IC50 = 31622.78 nM T05031 C4AGX5 122184531 IC50 = 31622.78 nM T05031 CQL4K5 122184532 IC50 = 12589.25 nM T05031 CX14YD 122184534 IC50 = 10000 nM T05031 CM6A4S 122184535 IC50 = 15848.93 nM T05031 CF86YS 122184536 IC50 = 25118.86 nM T05031 CH08SN 122184537 IC50 = 63095.73 nM T05031 CYRH97 122184538 IC50 = 50118.72 nM T05031 CD4W0Z 122184539 IC50 > 199526.23 nM T05031 CH8Y3Q 122184540 IC50 > 199526.23 nM T05031 CDA85R 122184541 IC50 > 199526.23 nM T05031 CF36XJ 122184542 IC50 > 199526.23 nM T05031 CQ6O7H 122184543 IC50 > 199526.23 nM T05031 CS4MN0 122184544 IC50 > 199526.23 nM T05031 CKT74G 122185265 IC50 = 47 nM T05031 CJ6C1O 122185267 IC50 = 41 nM T05031 CZE35C 122648343 IC50 > 10000 nM T05031 C54RNT 122648367 IC50 > 10000 nM T05031 C1UVI7 122648600 IC50 > 1000 nM T05031 CMX59K 122648648 IC50 = 34 nM T05031 CVZ64I 122648649 IC50 > 10000 nM T05031 CMG21L 122705987 IC50 = 5800 nM T05031 CW5EK9 122705988 IC50 = 5000 nM T05031 CPTY78 124518210 IC50 = 396 nM T05031 C98DKI 127025346 IC50 = 23 nM T05031 CBXJ67 127025628 IC50 = 9.4 nM T05031 CSV3R7 127029064 IC50 = 13 nM T05031 CGKR53 127032915 IC50 > 5000 nM T05031 C41YQI 127035981 IC50 > 5000 nM T05031 CRLD82 127039546 IC50 = 10000 nM T05031 C3ZXT2 127040693 IC50 = 3200 nM T05031 C6X0NR 127041034 IC50 > 10000 nM T05031 CLUK47 127042289 IC50 = 6900 nM T05031 C05MRE 127042767 IC50 = 3400 nM T05031 CG8DA9 127045861 IC50 = 5600 nM T05031 CVF8Z9 127045862 IC50 = 89 nM T05031 CA82TY 127045875 IC50 = 17 nM T05031 CH68NT 127046076 IC50 = 1120 nM T05031 CA2XD5 127046077 IC50 = 5290 nM T05031 C60UIQ 127046089 IC50 = 107 nM T05031 C9J1DA 127046090 IC50 = 197 nM T05031 COJ68G 127046117 IC50 = 10 nM T05031 C34REM 127046317 IC50 = 8 nM T05031 CIQO47 127046318 IC50 = 120 nM T05031 CC4ND8 127046862 IC50 = 3850 nM T05031 C0KE3Q 127046987 IC50 = 6 nM T05031 CY2P1X 127047138 IC50 = 3 nM T05031 CE2PM8 127047139 IC50 = 12 nM T05031 CZ2R0C 127047140 IC50 = 7 nM T05031 C6UYT9 127047141 IC50 = 4 nM T05031 CT89GI 127047683 IC50 = 6 nM T05031 CQ79JL 127047684 IC50 = 45 nM T05031 C7D0FN 127047685 IC50 = 10 nM T05031 CA87MN 127047796 IC50 = 5 nM T05031 CN94CQ 127047797 IC50 = 3 nM T05031 C3IC2Z 127052212 IC50 = 4073 nM T05031 CO8L3T 129029965 IC50 > 513 nM T05031 CX3WZ9 129029966 IC50 = 44 nM T05031 CN2D6Q 129029978 IC50 = 3 nM T05031 C1ZMP0 129029979 IC50 = 2 nM T05031 C02BTR 129030078 IC50 = 148 nM T05031 C4RW1X 129030093 IC50 = 6 nM T05031 C6T9RI 129030181 IC50 = 9 nM T05031 CY0BE9 129030296 IC50 = 2 nM T05031 C5GRU6 129030297 IC50 > 513 nM T05031 C7QYF2 129030298 IC50 = 1.35 nM T05031 C18NHD 130302549 IC50 <= 10000 nM T05031 CL13RZ 130302558 IC50 <= 10000 nM T05031 CF5JZ3 130302563 IC50 <= 10000 nM T05031 CD46EL 130302605 IC50 <= 10000 nM T05031 CNI8M6 130302620 IC50 <= 10000 nM T05031 CI6WN9 130302651 IC50 <= 10000 nM T05031 C5ZP0L 130302658 IC50 <= 10000 nM T05031 CW61SG 130302663 IC50 <= 10000 nM T05031 CB27ZG 130302668 IC50 <= 10000 nM T05031 C5VYM6 130302674 IC50 <= 10000 nM T05031 C0FQR2 130302675 IC50 <= 10000 nM T05031 CB34HQ 130302676 IC50 <= 10000 nM T05031 CQR1I8 130302685 IC50 <= 10000 nM T05031 C17DZF 130302698 IC50 <= 10000 nM T05031 CBC6W7 130302701 IC50 <= 10000 nM T05031 CBT21G 130302702 IC50 <= 10000 nM T05031 CDZ45O 130302703 IC50 <= 10000 nM T05031 C2GWU8 130302709 IC50 <= 10000 nM T05031 CV3M6Y 130302710 IC50 <= 10000 nM T05031 C39UQN 130302731 IC50 <= 10000 nM T05031 CL9O8X 130302732 IC50 <= 10000 nM T05031 CL69GM 130302740 IC50 <= 10000 nM T05031 CH8YK9 130302741 IC50 <= 10000 nM T05031 CQR2W9 130302781 IC50 <= 10000 nM T05031 C9HC8A 130302803 IC50 <= 10000 nM T05031 CIK25W 130302809 IC50 <= 10000 nM T05031 CI08PF 130332501 IC50 <= 10000 nM T05031 C1H4UT 130332505 IC50 <= 10000 nM T05031 CZPI64 130332579 IC50 <= 10000 nM T05031 CDS9F3 130332582 IC50 <= 10000 nM T05031 C3G0HF 130332585 IC50 <= 10000 nM T05031 CX13UC 130332620 IC50 <= 10000 nM T05031 CED6F3 130332657 IC50 <= 10000 nM T05031 C73KWM 130338615 IC50 = 55 nM T05031 C47CAY 130421765 IC50 > 31622.78 nM T05031 C84YKI 130422161 IC50 > 31622.78 nM T05031 CK68CA 130453737 IC50 = 10300 nM T05031 CUO41K 130470684 IC50 = 12800 nM T05031 CP32GB 132005220 IC50 > 10000 nM T05031 CUN18W 132005225 IC50 = 4800 nM T05031 CD84OI 132005228 IC50 = 540 nM T05031 C7ASP9 132005246 IC50 = 610 nM T05031 C4M8WN 132209922 IC50 = 795 nM T05031 CFI23B 132210082 IC50 = 1200 nM T05031 CH8DP7 132220479 IC50 > 5000 nM T05031 C6XZ4A 132271619 IC50 = 34 nM T05031 CH27LV 132271620 IC50 = 138 nM T05031 CCTK95 132271625 IC50 = 43 nM T05031 C4Q5LF 132471857 IC50 = 360 nM T05031 CJE34F 132597748 IC50 = 2200 nM T05031 CCV46G 132606879 IC50 = 158.49 nM T05031 CT2PN8 132990561 IC50 = 175 nM T05031 CG6M4F 134132862 IC50 = 2000 nM T05031 CFG90E 134132909 IC50 = 3880 nM T05031 CB86SC 134134086 IC50 = 2114 nM T05031 C4YNH0 134134126 IC50 = 669 nM T05031 C0EK8P 134134680 IC50 = 655 nM T05031 CLDS18 134135780 IC50 = 1400 nM T05031 CE12WX 134136190 IC50 = 955 nM T05031 C6IMP8 134136890 IC50 = 38 nM T05031 C0A1UM 134138053 IC50 = 956 nM T05031 C6OGM2 134138249 IC50 = 360 nM T05031 CQ2S4X 134138703 IC50 = 9010 nM T05031 CL3Q6G 134140420 IC50 = 1480 nM T05031 CTDG86 134140525 IC50 = 428 nM T05031 CDJ10M 134142931 IC50 = 1790 nM T05031 CUE85S 134143151 IC50 > 50000 nM T05031 CN59WG 134143270 IC50 = 540 nM T05031 CL4E9X 134144824 IC50 = 3210 nM T05031 CQ9G7H 134145670 IC50 = 1940 nM T05031 C1PVM6 134145863 IC50 > 10000 nM T05031 C6G8EJ 134146051 IC50 = 19000 nM T05031 CIPL93 134147099 IC50 = 1940 nM T05031 CBN10Y 134147858 IC50 = 554 nM T05031 C8ITR3 134147904 IC50 > 50000 nM T05031 CV2QA7 134148173 IC50 = 190 nM T05031 CXA3V0 134148445 IC50 > 9100 nM T05031 C3FO5C 134149163 IC50 = 3200 nM T05031 C0S8CM 134150384 IC50 = 52 nM T05031 CXU92M 134150578 IC50 = 860 nM T05031 CDA43X 134150949 IC50 = 521 nM T05031 CG8LE2 134151667 IC50 < 10000 nM T05031 CPX9K8 134152185 IC50 = 1210 nM T05031 CK43EY 134152988 IC50 = 3210 nM T05031 CE3C2V 134154007 IC50 = 1060 nM T05031 CL5MR8 134154147 IC50 = 1797 nM T05031 CS2QP7 134154582 IC50 = 304 nM T05031 CJDY92 134155338 IC50 = 811 nM T05031 CSK9Q8 134155414 IC50 = 1328 nM T05031 C2QGB3 134156160 IC50 = 1280 nM T05031 C42RJH 134157534 IC50 = 30 nM T05031 CJXA12 134611894 IC50 > 31622.78 nM T05031 CX0UR7 134694318 IC50 > 27000 nM T05031 C9FUK2 135151360 IC50 > 30000 nM T05031 CT0GQ6 135197577 IC50 = 1.2 nM T05031 C87VKA 135197594 IC50 = 1.1 nM T05031 CQXS07 135197635 IC50 = 0.4 nM T05031 C7KXF1 135197643 IC50 = 0.53 nM T05031 CY38TL 135391000 IC50 = 699.4 nM T05031 COG86Z 135397763 IC50 = 501.19 nM T05031 CWL67T 135397764 IC50 = 1000 nM T05031 CX8AI4 135398491 IC50 = 350 nM T05031 CH8TR5 135426721 IC50 = 14000 nM T05031 C6AZ2R 135435018 IC50 > 25118.86 nM T05031 C3QJ8W 135566371 IC50 = 697 nM T05031 C24ZGX 135566644 IC50 = 76 nM T05031 C2QDV5 135566741 IC50 = 42 nM T05031 C2UN0D 135742360 IC50 = 5800 nM T05031 CU29YK 135750268 IC50 = 380 nM T05031 C02PHA 135927892 IC50 = 25118.86 nM T05031 CS8T3D 135927897 IC50 > 25118.86 nM T05031 C12UDA 135947972 IC50 = 1450 nM T05031 CN42ZS 135947973 IC50 = 8600 nM T05031 CF8AO3 135947974 IC50 = 2530 nM T05031 CW08GJ 135947976 IC50 = 467 nM T05031 C8O9HG 135947977 IC50 = 100000 nM T05031 CJN7E2 135947978 IC50 = 2100 nM T05031 CFKH34 135947979 IC50 = 3200 nM T05031 C0ZH9X 135981194 IC50 > 100000 nM T05031 C4G2HP 135995897 IC50 = 80 nM T05031 CNF15Q 135995898 IC50 = 56 nM T05031 C98HZG 135995899 IC50 = 93 nM T05031 CIQ82W 135995900 IC50 = 67 nM T05031 CP1US5 136041737 IC50 = 17 nM T05031 CXH63V 136041747 IC50 = 30 nM T05031 C6B5TC 136041748 IC50 = 82 nM T05031 CU6XG1 136041749 IC50 = 85 nM T05031 C0U5DB 136041750 IC50 = 193 nM T05031 C48KAQ 136041752 IC50 = 49 nM T05031 C74PRL 136041753 IC50 = 26 nM T05031 CT4FJ1 136041757 IC50 = 4 nM T05031 CCS2G6 136041761 IC50 = 143 nM T05031 CEZP21 136041762 IC50 = 16 nM T05031 CJ58TD 136041764 IC50 = 88 nM T05031 CX67QW 136041765 IC50 = 8 nM T05031 CK0H2Q 136041766 IC50 = 105 nM T05031 CQP7B6 136041767 IC50 = 47 nM T05031 CM65BS 136041773 IC50 = 26 nM T05031 C6P7JB 136041775 IC50 = 63 nM T05031 C5CJF7 136041776 IC50 = 9 nM T05031 C3XIZ8 136041777 IC50 = 109 nM T05031 C32LKO 136041785 IC50 = 140 nM T05031 C90ARP 136041787 IC50 = 386 nM T05031 CZ3BN1 136041792 IC50 = 5 nM T05031 CG19DI 136041799 IC50 = 90 nM T05031 CXJA29 136041804 IC50 = 22 nM T05031 CHT31V 136041805 IC50 = 4 nM T05031 CO8C4J 136041817 IC50 = 12 nM T05031 C4QU6G 136041827 IC50 = 79 nM T05031 CNE10X 136041834 IC50 = 41 nM T05031 CS3AE1 136041847 IC50 = 13 nM T05031 CZC47Y 136041848 IC50 = 33 nM T05031 C7PHA5 136044403 IC50 = 1 nM T05031 CA91JG 136069599 IC50 = 8 nM T05031 CGAB91 136069600 IC50 = 33 nM T05031 C3ZAW2 136069605 IC50 = 9 nM T05031 C8JXL5 136069609 IC50 = 10 nM T05031 C9I0EQ 136069610 IC50 = 98 nM T05031 C25EYJ 136069611 IC50 = 17 nM T05031 C2S5QF 136069615 IC50 = 332 nM T05031 CI1LY8 136096349 IC50 = 1700 nM T05031 CC4UM3 136176116 IC50 = 10 nM T05031 CJRK81 136176117 IC50 = 26 nM T05031 C63IOS 136176118 IC50 = 17 nM T05031 C3KW7H 136176119 IC50 > 10000 nM T05031 C69AKQ 136176120 IC50 = 3410 nM T05031 CF17KO 136176121 IC50 = 125 nM T05031 CU3TE0 136176122 IC50 = 75 nM T05031 C6C5KB 136176123 IC50 = 233 nM T05031 C3X5KE 136176124 IC50 = 202 nM T05031 CA8C5E 136176125 IC50 = 127 nM T05031 C5OMG2 136176126 IC50 = 13 nM T05031 CP2YM7 136176127 IC50 = 90 nM T05031 C8XIJ0 136176128 IC50 = 22 nM T05031 CUY8N4 136176129 IC50 = 113 nM T05031 C3J4ME 136176130 IC50 = 44 nM T05031 CR1NZ2 136176131 IC50 = 47 nM T05031 C4WG2F 136176132 IC50 = 6 nM T05031 CJ8EC5 136176139 IC50 = 289 nM T05031 CQ84IZ 136180335 Ki > 4000 nM T05031 C1LK9U 136183381 IC50 = 1 nM T05031 C5EU1H 136188794 IC50 = 34000 nM T05031 C27TKQ 136196449 IC50 = 167 nM T05031 CC1X7G 136227360 IC50 = 1900 nM T05031 C5KW4P 136227361 IC50 = 63000 nM T05031 CK9S4X 136229137 IC50 = 93 nM T05031 CAI9M5 136229138 IC50 = 84 nM T05031 C8M5HN 136229139 IC50 = 470 nM T05031 C5ZFP8 136229140 IC50 = 570 nM T05031 CS1X6P 136229141 IC50 = 1400 nM T05031 CXQG23 136229142 IC50 = 1500 nM T05031 C07INE 136229143 IC50 = 34 nM T05031 CHXY59 136229144 IC50 = 24000 nM T05031 CVHL13 136229146 IC50 = 31000 nM T05031 CDEX74 136229147 IC50 = 7 nM T05031 CRJ47T 136229148 IC50 = 11000 nM T05031 C7S1YJ 136230225 IC50 = 142 nM T05031 C3Q6ED 136230226 IC50 = 81 nM T05031 CKPF02 136230227 IC50 = 236 nM T05031 CZY9O0 136230228 IC50 = 398 nM T05031 CRET01 136230229 IC50 = 15 nM T05031 CX1KI8 136230230 IC50 = 5 nM T05031 C3Z5MH 136230231 IC50 = 53 nM T05031 CUE6N8 136230232 IC50 = 6 nM T05031 C8Q1AP 136230233 IC50 = 2 nM T05031 C70RXE 136230234 IC50 = 3 nM T05031 C4W0KN 136230235 IC50 = 26 nM T05031 CMZN01 136230236 IC50 = 175 nM T05031 CCU0H5 136241428 IC50 = 5 nM T05031 C4QMY7 136244246 IC50 > 100000 nM T05031 CEU87Z 136245089 IC50 = 102 nM T05031 CL4MO3 136249382 IC50 = 17 nM T05031 C04LZP 136254186 IC50 > 100000 nM T05031 C8PT7R 136254187 IC50 = 13620 nM T05031 CCJV79 136254188 IC50 = 43670 nM T05031 C5QE8W 136254189 IC50 = 51750 nM T05031 C0GZV9 136254283 IC50 = 158 nM T05031 CMWA86 136264282 IC50 = 4 nM T05031 C1HI5T 136264454 IC50 = 1 nM T05031 CAL31Q 137167625 IC50 = 17 nM T05031 CG1MD6 137167628 IC50 = 48 nM T05031 CO3HE0 137167632 IC50 = 8 nM T05031 CX96FQ 137289808 IC50 = 11 nM T05031 CV3UE9 137333450 IC50 = 284 nM T05031 C7MR0T 137632022 IC50 = 1500 nM T05031 CIX4S7 137633081 IC50 = 100 nM T05031 C34MHP 137634951 IC50 = 317 nM T05031 C9GXM1 137635017 IC50 = 316.23 nM T05031 CO8X7R 137636042 IC50 = 76 nM T05031 CMN6T7 137636115 IC50 = 530 nM T05031 CMZV19 137639099 IC50 = 50.12 nM T05031 CS78JW 137639139 IC50 = 87 nM T05031 C4TSZ8 137639858 IC50 = 501.19 nM T05031 CA0QO6 137640453 IC50 = 509 nM T05031 CQ8X0E 137641383 IC50 > 15000 nM T05031 C0I6RQ 137641405 IC50 = 1000 nM T05031 C5X3TH 137642662 IC50 > 15000 nM T05031 CS18XW 137642670 IC50 = 16000 nM T05031 CP3JK1 137643598 IC50 = 1258.93 nM T05031 C5ERV3 137646413 IC50 = 1700 nM T05031 CZC27Y 137646667 IC50 = 100 nM T05031 C3TXN9 137647591 IC50 = 1650 nM T05031 C4Z0NQ 137648826 IC50 = 316.23 nM T05031 C37WLI 137650083 IC50 = 24 nM T05031 CHT1R8 137650579 IC50 = 398.11 nM T05031 CN78RE 137653565 IC50 = 125.89 nM T05031 C4N5LS 137655123 IC50 = 630.96 nM T05031 CTB78E 137655854 IC50 = 32 nM T05031 CJB90Y 137656872 IC50 = 1300 nM T05031 CE9H8D 137657006 IC50 = 398.11 nM T05031 C41OPW 137658031 IC50 = 794.33 nM T05031 C6BF8E 137658458 IC50 > 15000 nM T05031 CCP6G3 137659846 IC50 = 1.4 nM T05031 CP5K4E 137660883 IC50 = 2020 nM T05031 C1OLQ3 137660961 IC50 = 1258.93 nM T05031 CM6FS2 137661095 IC50 = 158.49 nM T05031 C8R3JK 137661301 IC50 = 50.12 nM T05031 CA3C4O 138454792 IC50 = 101 nM T05031 CKDZ26 138504497 IC50 = 8100 nM T05031 C0BFS3 139327957 IC50 = 214 nM T05031 C7ZAQ1 141406387 IC50 = 54870 nM T05031 C7NUI8 141406388 IC50 = 67920 nM T05031 CQYI18 141406390 IC50 = 18660 nM T05031 CUA1D0 141406392 IC50 = 32650 nM T05031 CP0R6Y 141406393 IC50 = 1680 nM T05031 C1EVQ0 141406394 IC50 = 20840 nM T05031 C2QP0F 141406396 IC50 = 22650 nM T05031 CY2M0B 141406399 IC50 = 9580 nM T05031 CC3OU2 141406400 IC50 = 56740 nM T05031 CKV13Y 141406404 IC50 = 22840 nM T05031 C3Q1VL 141419885 IC50 = 263.8 nM T05031 C3EJX8 141419888 IC50 = 584.5 nM T05031 CKX4P3 141446054 IC50 = 25118.86 nM T05031 C4C0QL 141461656 IC50 = 29 nM T05031 CZV17F 141461667 IC50 = 4 nM T05031 CD5VE0 141461669 IC50 = 6 nM T05031 CU6LE4 141461671 IC50 = 39 nM T05031 CV54CS 141471198 IC50 = 3.4 nM T05031 C25HYI 141471200 IC50 = 1.2 nM T05031 CZS03J 141509623 IC50 = 838 nM T05031 C1R9AN 141518981 IC50 = 89 nM T05031 C4MH5U 141518989 IC50 = 106 nM T05031 CQT27N 141520958 IC50 = 108 nM T05031 CU03GW 142506036 IC50 = 188 nM T05031 C74MXW 142506065 IC50 = 33 nM T05031 CX6BQ7 142506102 IC50 = 26 nM T05031 CY3BM0 142506119 IC50 = 5210 nM T05031 CC6MD0 142506155 IC50 = 279 nM T05031 CT3U9R 142506192 IC50 = 12 nM T05031 C1T3IQ 142506210 IC50 = 286 nM T05031 C1U3CA 142506238 IC50 = 842 nM T05031 C7QMG9 145108300 IC50 = 6.6 nM T05031 C1FIE4 145439085 IC50 = 1482 nM T05031 CI40JE 145951013 IC50 = 317.1 nM T05031 C6YT8E 145951131 IC50 = 8940 nM T05031 CFW62M 145951569 IC50 = 98.8 nM T05031 CHA84K 145951830 IC50 = 8769 nM T05031 CT4I9A 145952160 IC50 = 23.4 nM T05031 C91GVH 145952598 IC50 = 7.3 nM T05031 C1W0GJ 145952796 IC50 > 25118.86 nM T05031 CVMF13 145953272 IC50 > 10000 nM T05031 CYL5T1 145953372 IC50 <= 10000 nM T05031 CP14AV 145953653 IC50 = 57.2 nM T05031 CY8D5Q 145953886 IC50 = 307.5 nM T05031 C3ZUW8 145954195 IC50 = 148.5 nM T05031 C1NJB7 145955070 IC50 = 19.5 nM T05031 CRHE01 145955133 IC50 <= 10000 nM T05031 C7MP9Z 145955279 IC50 = 82.1 nM T05031 C7K8VT 145955565 IC50 = 62.5 nM T05031 CPU4X2 145955670 IC50 = 766.4 nM T05031 C3ST5Y 145955693 IC50 = 92.3 nM T05031 C1VH5X 145955836 IC50 = 124.2 nM T05031 C7K2YF 145956631 IC50 <= 10000 nM T05031 CQW74M 145956683 IC50 = 34.7 nM T05031 CJ1F6A 145956725 IC50 = 228.8 nM T05031 C12IFO 145956886 IC50 = 119.3 nM T05031 C9O2PL 145958063 IC50 = 155.9 nM T05031 CQH01X 145958257 IC50 <= 10000 nM T05031 C3DGU7 145958571 IC50 = 50 nM T05031 C9NS6T 145958690 IC50 = 243.7 nM T05031 C7ZO9V 145959196 IC50 = 1539 nM T05031 CSC81H 145959429 IC50 = 27.5 nM T05031 C0S1YM 145959980 IC50 = 290 nM T05031 CT3I2R 145960112 IC50 = 84.2 nM T05031 C8MJ9X 145960272 IC50 = 109.3 nM T05031 C50URO 145960355 IC50 = 7 nM T05031 CF36RA 145961004 IC50 = 28.4 nM T05031 CHF56O 145961403 IC50 > 9100 nM T05031 C2GT9Y 145961404 IC50 > 9100 nM T05031 CAI0D6 145963117 IC50 = 386 nM T05031 CU9XC4 145966764 IC50 = 3 nM T05031 C97IKW 145969580 IC50 = 220.3 nM T05031 CK82QG 145969816 IC50 = 4936 nM T05031 C71YAK 145970017 IC50 = 355000 nM T05031 CZ98FH 145971490 IC50 = 1761 nM T05031 CTB97Z 145971948 IC50 = 480.5 nM T05031 CGQJ04 145972017 IC50 = 422.1 nM T05031 C96IUM 145973569 IC50 = 2 nM T05031 CZ9G6E 145974533 IC50 = 201.5 nM T05031 C3LR4O 145976442 IC50 = 9412 nM T05031 C3YG4Z 145977475 IC50 = 2 nM T05031 CPZS56 145982349 EC50 = 5700 nM T05031 CH90CT 145983168 IC50 = 382.3 nM T05031 CJU02I 145983624 IC50 = 6955 nM T05031 CVS2U0 145983808 IC50 = 3369 nM T05031 CF8MR5 145986347 IC50 = 430000 nM T05031 C6XMQ8 145989163 EC50 = 3340 nM T05031 C8X2IT 145996536 IC50 > 10000 nM T05031 C6RPG0 146014481 IC50 = 288.4 nM T05031 CI85VS 146731761 IC50 = 120 nM T05031 C4MC0S 149169124 IC50 = 2490 nM T05031 CVW62P 149242889 IC50 = 4640 nM T05031 CN87RZ 149370890 IC50 = 850 nM T05031 CK4FJ1 149556361 IC50 = 5750 nM T05031 C8UQL4 153940691 IC50 = 2650 nM T05031 CMZ68Q 153940692 IC50 = 210 nM T05031 C5X7JK 154734328 IC50 = 2511.89 nM T05031 CDT8F2 155510913 IC50 = 3981.07 nM T05031 CZJ9D6 155512258 IC50 = 59 nM T05031 CG9I4X 155512515 IC50 = 410 nM T05031 CR1Z8A 155512529 IC50 > 10000 nM T05031 CQZY50 155512775 IC50 = 398.11 nM T05031 C5V2GO 155512947 IC50 = 3981.07 nM T05031 C1DIT4 155513047 IC50 = 1584.89 nM T05031 C8PG6Z 155513084 IC50 = 2511.89 nM T05031 C5M6NS 155513226 IC50 = 15300 nM T05031 C45SYX 155513615 IC50 = 16 nM T05031 CBH57O 155514764 IC50 = 2511.89 nM T05031 C5C9EG 155515047 IC50 = 5011.87 nM T05031 CEFS61 155515135 IC50 = 2190 nM T05031 C0AXF7 155515394 IC50 = 6309.57 nM T05031 C7Q3FR 155515734 IC50 = 6309.57 nM T05031 C30ZFN 155516445 IC50 = 10000 nM T05031 CJDG04 155516604 IC50 = 1995.26 nM T05031 CYO19V 155517071 IC50 = 1995.26 nM T05031 CYWX76 155517213 IC50 = 7943.28 nM T05031 C4G8YN 155517534 IC50 = 342 nM T05031 CW7OM6 155518918 IC50 = 513 nM T05031 CC51GM 155519635 IC50 = 1995.26 nM T05031 CQEK39 155520373 IC50 = 5 nM T05031 C5D6YX 155521099 IC50 > 10000 nM T05031 CEA3M1 155521494 IC50 = 398.11 nM T05031 CBSR95 155522042 IC50 = 11320 nM T05031 CZO7Q8 155522149 IC50 = 601 nM T05031 CCGW06 155523124 IC50 = 10000 nM T05031 C4TLQ7 155523447 IC50 > 10000 nM T05031 CZG27I 155523570 IC50 = 342 nM T05031 C37RVF 155523599 IC50 = 2040 nM T05031 C4H2AB 155524238 IC50 = 630.96 nM T05031 CP18VT 155524467 IC50 = 1000 nM T05031 CUP7L2 155524901 IC50 = 3162.28 nM T05031 C2BL5I 155525312 IC50 = 1000 nM T05031 C10RZQ 155525477 IC50 = 630.96 nM T05031 CF76OV 155525717 IC50 = 31.4 nM T05031 C0UA4D 155525996 IC50 = 794.33 nM T05031 C3EAR8 155526323 IC50 = 1995.26 nM T05031 C82NUW 155527501 IC50 = 166 nM T05031 CK07GS 155527559 IC50 = 217 nM T05031 CX12MK 155527651 IC50 = 159 nM T05031 C8Z3TK 155528581 IC50 = 1584.89 nM T05031 C0B2NV 155528644 IC50 = 8050 nM T05031 C9L6OC 155529247 IC50 = 279 nM T05031 C2FE1S 155529479 IC50 = 398.11 nM T05031 CB90AR 155529643 IC50 = 158.49 nM T05031 CFV1S0 155529706 IC50 = 207 nM T05031 C14QOF 155530163 IC50 = 630.96 nM T05031 C4I5UP 155530224 IC50 = 1000 nM T05031 CX6N3Y 155531155 IC50 = 501.19 nM T05031 C9AXO7 155531257 IC50 = 6309.57 nM T05031 CDI4V8 155531526 IC50 = 24 nM T05031 CE6QP1 155532037 IC50 = 125.89 nM T05031 CIM18N 155532540 IC50 = 8900 nM T05031 C3XFB8 155532820 IC50 = 158.49 nM T05031 CIYA39 155532858 IC50 = 766 nM T05031 C0GR1J 155533050 IC50 = 9.1 nM T05031 CQS8P1 155533070 IC50 = 3981.07 nM T05031 C0SZR9 155533335 IC50 = 7943.28 nM T05031 CAT9V1 155533370 IC50 = 4270 nM T05031 C67ERP 155533384 IC50 = 1584.89 nM T05031 CL8OM7 155533564 IC50 = 60 nM T05031 CBM24U 155533579 IC50 = 1995.26 nM T05031 CR5H8B 155533591 IC50 = 1995.26 nM T05031 CA7T0Y 155533911 IC50 > 10000 nM T05031 CN1ST4 155534269 IC50 = 398.11 nM T05031 CBEG39 155534594 IC50 = 2511.89 nM T05031 CTZ3E0 155534905 IC50 = 169 nM T05031 CN6KJ5 155535520 IC50 = 1258.93 nM T05031 C5F2TY 155535537 IC50 = 3162.28 nM T05031 CKB2U4 155535691 IC50 = 630.96 nM T05031 CY7X3M 155535740 IC50 = 630.96 nM T05031 C70UDF 155536179 IC50 = 6309.57 nM T05031 CEJ6L1 155536226 IC50 = 147.4 nM T05031 CNB24M 155536473 IC50 = 1258.93 nM T05031 C2CG1A 155537016 IC50 = 794.33 nM T05031 C8AJ6C 155538256 IC50 = 150.1 nM T05031 CQ1E6H 155538266 IC50 = 316.23 nM T05031 CZ19AN 155538609 IC50 = 329 nM T05031 CHR8M1 155538990 IC50 > 10000 nM T05031 CC1BG2 155539321 IC50 > 10000 nM T05031 CF20PS 155539394 IC50 = 1000 nM T05031 C8LKW4 155540264 IC50 = 2511.89 nM T05031 CKBW37 155542030 IC50 = 3990 nM T05031 C8OC2P 155542800 IC50 = 3200 nM T05031 CVNR95 155542898 IC50 = 536 nM T05031 C1SY0G 155543154 IC50 = 15600 nM T05031 CZY0N4 155543588 IC50 = 379 nM T05031 CJB8C9 155543659 IC50 = 215 nM T05031 CX1C8I 155544561 IC50 > 10000 nM T05031 CBN29V 155544583 IC50 = 139 nM T05031 C98FXC 155544955 IC50 = 775 nM T05031 CTSW53 155546042 IC50 > 10000 nM T05031 CQ6J7U 155546361 IC50 = 900 nM T05031 C8SQA2 155546999 IC50 = 251.19 nM T05031 CI6KO7 155548518 IC50 = 3981.07 nM T05031 CL4F8P 155549003 IC50 = 251.19 nM T05031 C4PEJ5 155549895 IC50 = 9710 nM T05031 CFP94J 155550309 IC50 = 3162.28 nM T05031 CQ5OD0 155550395 IC50 = 21 nM T05031 CK1JR7 155551961 IC50 = 5.6 nM T05031 CJ75BO 155552100 IC50 = 2140 nM T05031 CL04BD 155554125 IC50 = 300 nM T05031 CX9C6O 155554180 IC50 = 1000 nM T05031 CC13QL 155555170 IC50 = 1722 nM T05031 C2OGW1 155555483 IC50 = 162 nM T05031 CRO5Z3 155556073 IC50 = 146 nM T05031 CH2P4T 155556124 IC50 > 50118.72 nM T05031 CIU29Z 155556576 IC50 = 5400 nM T05031 CM3LI6 155556593 IC50 = 3358 nM T05031 CZ8CX1 155556887 IC50 = 1995.26 nM T05031 CG2FS6 155557123 IC50 = 2511.89 nM T05031 CFS63H 155557182 IC50 = 3540 nM T05031 C0FE4G 155557988 IC50 = 2821 nM T05031 CR8J0E 155558167 IC50 = 501.19 nM T05031 C52TSP 155558262 IC50 = 602 nM T05031 CS70ER 155559192 IC50 = 428 nM T05031 CVG49I 155560688 IC50 = 4140 nM T05031 C5S7AL 155560766 IC50 = 1995.26 nM T05031 CLO3B1 155561152 IC50 = 1910 nM T05031 C8XS0L 155561165 IC50 = 1258.93 nM T05031 C72CQG 155561233 IC50 = 630.96 nM T05031 C1INL7 155561328 IC50 = 2511.89 nM T05031 CX6U2T 155562388 IC50 = 3981.07 nM T05031 CCF4W2 155563986 IC50 = 2511.89 nM T05031 CHK4E8 155565269 IC50 = 3162.28 nM T05031 C7PXA0 155565551 IC50 = 501.19 nM T05031 CY4N7O 155565715 IC50 = 15848.93 nM T05031 CVQ6Z4 155565763 IC50 = 6309.57 nM T05031 CMK4I3 155565845 IC50 = 1258.93 nM T05031 C59VPW 155565958 IC50 = 1995.26 nM T05031 CAP9F2 155566187 IC50 = 273 nM T05031 CM7E2G 155566279 IC50 = 1995.26 nM T05031 C9KQW3 155567372 IC50 = 2570 nM T05031 C1HQ5J 155568324 IC50 = 1554 nM T05031 CLA46O 155568356 IC50 = 1130 nM T05031 C7SLR8 155568452 IC50 = 1584.89 nM T05031 C1S8ZB 155568922 IC50 = 5740 nM T05031 C14LVO 155569074 IC50 = 1995.26 nM T05031 CFWP17 155569113 IC50 = 6237 nM T05031 CUH38L 155569363 IC50 = 9140 nM T05031 C4H0NE 155569598 IC50 = 7943.28 nM T05031 D00HSJ 10275789 IC50 = 340 nM T05031 D00ZIK 9908783 IC50 = 16000 nM T05031 D03EHM 24905142 IC50 = 1400 nM T05031 D03QQH 16760391 IC50 = 3700 nM T05031 D05USL 5278396 IC50 = 133 nM T05031 D06DNH 9907093 IC50 = 22 nM T05031 D06HVH 54613583 IC50 = 8600 nM T05031 D06PWI 42623951 IC50 = 1000 nM T05031 D07PMP 44187953 IC50 = 7 nM T05031 D08NQM 5289247 IC50 = 270 nM T05031 D0H2CM 135565635 IC50 = 2200 nM T05031 D0P5TI 58441401 IC50 = 166 nM T05031 D0R0TW 11964036 IC50 = 0.5 nM T05031 D0R2UG 52936849 IC50 = 59 nM T05031 D0S5YV 6852167 IC50 = 590 nM T05031 D0W8XH 9884685 IC50 = 3 nM T05031 D0Y3OO 11327430 IC50 = 16 nM T36725 D05WSP 11241908 Ki = 206 nM T36725 CJ6MK1 644475 Ki = 67200 nM T36725 C8VOM5 647799 Ki = 9100 nM T36725 CC13RQ 649517 Ki = 23900 nM T36725 CJ3DY5 655772 Ki = 292000 nM T36725 CE49ZA 856409 Ki = 7500 nM T36725 CS7GP6 861652 Ki = 14700 nM T36725 CT28UZ 1071864 Ki = 11600 nM T36725 CQGA28 1134678 Ki = 11700 nM T36725 C6LS4W 1154599 Ki = 7400 nM T36725 C0CSV5 1155310 Ki = 40000 nM T36725 C2Q0GS 1177046 Ki = 16600 nM T36725 CP1KV5 1374428 Ki = 4900 nM T36725 CLT49U 1429411 Ki = 364000 nM T36725 CEA19S 1442054 Ki = 25900 nM T36725 CKU3V9 1451696 Ki = 25100 nM T36725 CAJM89 1457216 Ki = 74500 nM T36725 C3QL6D 1463403 Ki = 1200 nM T36725 CEL50A 3173507 Ki = 4500 nM T36725 C34COQ 3189957 Ki = 23000 nM T36725 CI37KJ 3190690 Ki = 10800 nM T36725 CFC46P 5770758 Ki = 15000 nM T36725 C40BDL 9834739 IC50 = 20 nM T36725 CF5A3T 9837547 IC50 = 70 nM T36725 CV6F0Y 9900049 IC50 = 160 nM T36725 CHI95J 9926432 IC50 = 4 nM T36725 C39EUV 10149451 Ki = 240 nM T36725 C5G7KU 10308323 Ki = 265 nM T36725 C1GUQ8 10929000 Ki = 3000 nM T36725 CRH61B 10951188 Ki = 1060 nM T36725 C21DFC 10994303 Ki = 9100 nM T36725 CXT3L1 11149158 Ki = 1160 nM T36725 CY97KP 11494236 Ki = 70000 nM T36725 C5Q6GR 11537817 Ki = 410000 nM T36725 C9Y2IN 11731059 Ki = 3900 nM T36725 CAYN20 21303381 Ki > 10000 nM T36725 C3PI9L 21604546 Ki = 400000 nM T36725 C2ZV4R 22289844 Ki = 2720 nM T36725 CUY0G8 25110755 IC50 = 360 nM T36725 C05QKN 44308084 IC50 = 600 nM T36725 C1HCY9 44308186 IC50 = 1500 nM T36725 CD7IK4 44308237 IC50 = 1 nM T36725 C9IPN5 44308238 IC50 = 150 nM T36725 CBR39F 44308352 IC50 = 4 nM T36725 CH27SZ 44308370 IC50 = 1 nM T36725 C5LY4T 44308385 IC50 = 1 nM T36725 C5JY4E 44585289 Ki = 15100 nM T36725 CR42OD 44585290 Ki = 16700 nM T36725 CM4NI0 44585291 Ki = 9700 nM T36725 C8Z6MS 44585292 Ki = 7200 nM T36725 CRSD61 44585293 Ki = 9200 nM T36725 CU73FS 44585298 Ki = 23500 nM T36725 CSLH24 44585299 Ki = 16700 nM T36725 CO9W4X 44592983 Ki = 500000 nM T36725 C1F4ZM 44592984 Ki = 43000 nM T36725 CQ8T9I 44593009 Ki = 275000 nM T36725 C0BR9X 45268420 Ki = 33600 nM T36725 CHU74W 45270941 Ki = 196000 nM T36725 CUFH15 45272673 Ki = 20800 nM T36725 CZY78Q 46225030 Ki = 238 nM T36725 CEQ39A 46225031 Ki = 49 nM T36725 CITR87 46225064 Ki = 27 nM T36725 CQH24P 46225065 Ki = 360 nM T36725 CB3ZI1 46225066 Ki > 10000 nM T36725 CMI2O3 59187303 IC50 = 190 nM T36725 CS49EB 112499887 Ki = 0.12 nM T36725 C0H8AW 122177723 IC50 = 1 nM T36725 D00GOD 10035600 IC50 = 3700 nM T36725 D06LNX 3858 Ki = 10000 nM T36725 D07RXJ 1438175 Ki = 20700 nM T36725 D08SBS 3464 Ki = 1100 nM T36725 D0O3QJ 10286113 Ki = 27 nM T69128 D03ZBT 11626560 Ki = 0.6 nM T69128 D04LVK 57379345 Ki = 0.4 nM T69128 D08PIE 68165256 IC50 = 1.9 nM T69128 D0AF6O 71731823 Ki < 0.02 nM T69128 D0R3JB 4212 IC50 = 2998.7 nM T69128 D0U3SY 49806720 Ki = 2000 nM T69128 D03HUX 49792852 IC50 > 10000 nM T69128 D03LWG 53235510 IC50 = 3263 nM T69128 D05NFR 135565923 IC50 = 8.4 nM T69128 D0D1GF 42642645 Ki = 8.2 nM T69128 D0E3TC 44259 IC50 = 0.07 nM T69128 D0O0LS 25141092 IC50 = 5 nM T69128 D0O9PQ 57390074 IC50 = 1.9 nM T69128 D03BNU 59604787 IC50 > 10000 nM T69128 D0T3ME 156422 IC50 > 30000 nM T69128 CACS26 11561968 Ki > 2000 nM T69128 CU0E8O 11690457 Ki > 2000 nM T69128 CUT5I7 44517769 IC50 = 1.7 nM T69128 CP9VW3 44626349 IC50 = 209 nM T69128 CLS29B 46872626 IC50 > 10000 nM T69128 C2Y6QS 50938552 IC50 > 10000 nM T69128 C9NYP4 51036677 IC50 > 10000 nM T69128 C4WRY3 51037112 IC50 > 10000 nM T69128 CRI28Z 51037948 IC50 > 10000 nM T69128 CEQN27 52936621 Ki > 1000 nM T69128 CM24LF 52938983 IC50 < 1 nM T69128 C8NA4L 53384644 IC50 > 30000 nM T69128 C1EVX0 58063117 IC50 = 15200 nM T69128 C1MR8Q 60097495 IC50 > 1000 nM T69128 CV63UL 67240318 IC50 > 10000 nM T69128 CCN01X 71547862 IC50 > 10000 nM T69128 CEV53L 71548006 IC50 = 43 nM T69128 CPG3A5 86302574 IC50 = 2829 nM T69128 CFB75T 90479825 IC50 = 124 nM T69128 CY0UC4 90645194 IC50 > 10000 nM T69128 CN64BI 102140478 IC50 = 13.6 nM T69128 CY7BI2 118706214 IC50 > 10000 nM T69128 C7Z3NM 118706420 IC50 = 59.1 nM T69128 C8GYA7 118706421 IC50 = 108 nM T69128 CHL9W3 118706422 IC50 = 63.8 nM T69128 C0E1JR 118706423 IC50 = 241 nM T69128 CK61DC 118706424 IC50 = 104 nM T69128 C5Y1GH 118706425 IC50 = 74.2 nM T69128 C71PFB 118706426 IC50 = 138 nM T69128 CE3KO4 118706427 IC50 = 283 nM T69128 CO1IL5 118706428 IC50 = 86.5 nM T69128 C4DH0Q 118706429 IC50 = 133 nM T69128 C6PTS1 118706430 IC50 = 105 nM T69128 CP2TO4 118706431 IC50 = 91.5 nM T69128 C9FRU1 118706432 IC50 = 56.6 nM T69128 CIGK87 118706433 IC50 = 25.4 nM T69128 C4I9KZ 118706553 IC50 = 139 nM T69128 CXWN35 118726561 IC50 = 920 nM T69128 CW4O3Q 118726562 IC50 = 119 nM T69128 CO8YT9 118726563 IC50 = 56 nM T69128 C3CSO5 118726564 IC50 = 57600 nM T69128 C9PW5V 118726565 IC50 = 88 nM T69128 CIJ1S2 118726566 IC50 = 780 nM T69128 CI50GB 118726567 IC50 = 108 nM T69128 CW7U2O 118726568 IC50 = 24 nM T69128 CCK37S 118726569 IC50 = 478 nM T69128 C5PX2O 118726570 IC50 = 55500 nM T69128 C9NPH1 118726571 IC50 = 1330 nM T69128 C38EYR 118726572 IC50 = 357 nM T69128 CLH5M3 118726575 IC50 = 570 nM T69128 CN35BC 118726576 IC50 = 330 nM T69128 C1WPB8 118726577 IC50 = 1250 nM T69128 C41LKS 118726578 IC50 = 6250 nM T69128 C08KEM 122179540 IC50 = 300 nM T69128 C3AJ4C 122179546 IC50 = 600 nM T69128 CG0RP7 122179547 IC50 = 60 nM T69128 C1A0SQ 122179548 IC50 = 210 nM T69128 CKS28E 127034802 IC50 > 1000 nM T69128 CUO0C5 132156633 IC50 > 10000 nM T69128 CPJG85 134135151 IC50 = 5.8 nM T69128 C9FZ3A 134136788 IC50 = 2.3 nM T69128 CG92RQ 134137314 IC50 = 3.4 nM T69128 C1U2MV 134137679 IC50 = 5 nM T69128 CHL7B1 134140023 IC50 = 2.7 nM T69128 C6M9DN 134140179 IC50 = 1.8 nM T69128 C8KC5F 134142230 IC50 = 5.5 nM T69128 CDCJ80 134148182 IC50 = 4.7 nM T69128 CZ8W6R 134612705 IC50 = 1.1 nM T69128 C25ERN 137631967 IC50 = 168.5 nM T69128 C06JRX 137637094 IC50 > 1000 nM T69128 C1DK0P 137651391 IC50 > 1000 nM T69128 CV5H3Z 137657932 IC50 = 272.9 nM T69128 CT1D9K 138454747 IC50 = 2300 nM T69128 COG63R 141482475 IC50 = 2400 nM T69128 CKN4Z9 141482476 IC50 > 10000 nM T69128 C1QZK2 141482477 IC50 = 9100 nM T69128 CX2TB0 141482479 IC50 = 1400 nM T69128 CFH6E9 141482480 IC50 = 6200 nM T69128 CWQ92I 141482481 IC50 = 2300 nM T69128 C16ZIH 141482484 IC50 = 1500 nM T69128 CPH01I 141482485 IC50 = 8700 nM T69128 C15RML 141482486 IC50 = 9400 nM T69128 CNR57A 141482487 IC50 = 570 nM T69128 C5GEQ3 141482489 IC50 = 1800 nM T69128 C0FG1K 141482490 IC50 = 2400 nM T69128 C0UIW1 141482492 IC50 = 370 nM T69128 CH9I3U 141482493 IC50 = 8400 nM T69128 C2DF4X 141482494 IC50 > 10000 nM T69128 CFE08V 141482495 IC50 > 10000 nM T69128 CJ61MC 141482496 IC50 > 10000 nM T69128 C34QYJ 141482498 IC50 = 2400 nM T69128 CC21GM 141482499 IC50 > 10000 nM T69128 C25PAE 141482501 IC50 = 9400 nM T69128 CQF23C 141482502 IC50 > 10000 nM T69128 CSK43T 141482503 IC50 > 10000 nM T69128 C0IBX2 141482504 IC50 = 440 nM T69128 CSD1Z6 141488410 IC50 = 1260 nM T69128 CVA4W1 141488417 IC50 = 7300 nM T69128 C1AL7N 145949714 IC50 = 440 nM T69128 CDZK73 145950618 IC50 > 10000 nM T69128 C6HC2M 145950676 IC50 = 7400 nM T69128 CBT87I 145950891 IC50 = 6300 nM T69128 CQ2I5Y 145951801 IC50 = 1800 nM T69128 CM3CX8 145952650 IC50 = 8 nM T69128 C8V4MP 145952681 IC50 = 3 nM T69128 COA5Y3 145953378 IC50 = 9.8 nM T69128 C8LMR5 145953442 IC50 > 10000 nM T69128 C89RPH 145954372 IC50 = 4.6 nM T69128 CA10CB 145954622 IC50 = 410 nM T69128 CV9M0Z 145955839 IC50 = 8700 nM T69128 C2V8DA 145957160 IC50 = 13.4 nM T69128 C2O1TV 145957224 IC50 = 9600 nM T69128 C0O3PM 145958131 IC50 > 10000 nM T69128 C42ZQH 145958534 IC50 = 19.3 nM T69128 CXWH23 145958592 IC50 = 8.5 nM T69128 C3TLJ8 145959766 IC50 > 10000 nM T69128 CI6C4A 145973385 IC50 = 640 nM T69128 C4X8LC 145979928 IC50 = 1600 nM T69128 CNFJ75 145980559 IC50 = 2000 nM T69128 CAE5G0 145987157 IC50 = 3400 nM T69128 C1J5IX 145990848 IC50 = 4600 nM T69128 C5KB0A 145991472 IC50 = 6100 nM T69128 CGA41L 146014467 IC50 = 530 nM T69128 C4PT8S 155511865 Ki < 0.07 nM T69128 CR68FM 155519610 IC50 = 0.81 nM T69128 CNU28S 155519814 IC50 = 0.97 nM T69128 CSRV18 155524183 IC50 > 10000 nM T69128 C4GR6U 155524577 IC50 = 3390 nM T69128 CE5U8Z 155526528 IC50 = 1210 nM T69128 CHI54P 155529236 IC50 = 3.2 nM T69128 C6VQ0W 155530641 IC50 = 1.7 nM T69128 CX7I1V 155531079 IC50 = 6.8 nM T69128 CVBK76 155531967 IC50 = 5.3 nM T69128 CGVZ73 155532854 IC50 = 1.7 nM T69128 CX91EL 155534287 IC50 = 2260 nM T69128 CM0U3I 155534552 IC50 = 0.43 nM T69128 CX3AU5 155534611 IC50 = 1080 nM T69128 CEQJ52 155534874 IC50 = 4.4 nM T69128 C78MZC 155536330 IC50 = 2 nM T69128 CRV8K0 155538035 IC50 > 10000 nM T69128 C80DML 155541340 IC50 > 10000 nM T69128 CL6A7R 155541437 IC50 = 12150 nM T69128 CT02GE 155541767 IC50 = 0.97 nM T69128 C60YKA 155548301 IC50 = 5.3 nM T69128 CZ4J2P 155552610 IC50 = 3.7 nM T69128 CS4RB8 155557858 IC50 = 2.3 nM T69128 C1OI5K 155559863 IC50 = 0.73 nM T69128 C1ZX4J 155563060 IC50 = 0.76 nM T69128 CJN3Q9 155564067 IC50 > 10000 nM T69128 D0K5UF 72710568 Ki = 0.02 nM T69128 D0R2WK 16038120 IC50 = 2 nM T95399 D0B3HD 2519 IC50 = 114000 nM T95399 D0LF1U 5287969 IC50 = 1000 nM T95399 C8IJ0B 79025 Ki = 1700000 nM T95399 C8WA2E 3658622 IC50 ~ 100000 nM T95399 C8BDA7 4369162 Ki = 5100 nM T95399 C0E9MB 9840862 IC50 = 14 nM T95399 CWS9P8 9931451 IC50 = 6000 nM T95399 CDZ2L0 9953189 IC50 = 50000 nM T95399 COL4X7 9954417 IC50 = 60 nM T95399 C65DJK 9958633 IC50 = 11 nM T95399 C5BAT1 10043666 IC50 = 55 nM T95399 CC4IR6 10125909 IC50 = 38 nM T95399 CA3TJ8 10409816 IC50 = 50000 nM T95399 CZR8W9 10477826 IC50 = 138 nM T95399 C8V9TB 11187969 IC50 = 120 nM T95399 CMI72Q 11200159 IC50 = 190 nM T95399 CL4JZ8 11200978 IC50 > 200000 nM T95399 CXRG64 11222164 IC50 = 110 nM T95399 C3C2JH 11292222 IC50 = 110 nM T95399 C1VH7I 11324538 IC50 = 2500 nM T95399 C1W7PG 11337343 IC50 = 200 nM T95399 CKZ57R 11338774 IC50 = 140 nM T95399 CW3C9Z 11451272 IC50 = 710 nM T95399 CXH6R7 11465977 IC50 = 350 nM T95399 CY0IT9 11475200 IC50 = 280 nM T95399 CKO62P 11475654 IC50 = 320 nM T95399 CP0XI8 11772828 IC50 = 730 nM T95399 CP56TC 11774080 IC50 = 190 nM T95399 CUC7N2 11785069 IC50 = 420 nM T95399 CY1J3I 13908996 Ki = 1000000 nM T95399 CI0JH1 19002057 Ki = 1.6 nM T95399 CDM7V9 21974595 IC50 = 32 nM T95399 CIK5V6 44342320 IC50 = 41 nM T95399 COZG47 44342348 IC50 = 12.9 nM T95399 C49TDU 44342362 IC50 = 52 nM T95399 CF8D0Y 44342363 IC50 = 15000 nM T95399 C30MEI 44342377 IC50 = 1195 nM T95399 CASE46 44342459 IC50 = 178 nM T95399 C25DBF 44342460 IC50 = 8.28 nM T95399 CQH1X0 44342462 IC50 = 10.61 nM T95399 CX2G3N 44342474 IC50 = 29 nM T95399 CNX08S 44342475 IC50 = 10 nM T95399 CXEC30 44342489 IC50 = 37 nM T95399 CK84CQ 44342512 IC50 = 91 nM T95399 C6M3LQ 44342540 IC50 = 185 nM T95399 C5R3WV 44342585 IC50 = 233 nM T95399 CA3G4I 44342602 IC50 = 6 nM T95399 CX15TC 44342751 IC50 = 26 nM T95399 CLZD72 44342773 IC50 = 19.9 nM T95399 CT1GA3 44345051 Ki = 11 nM T95399 CDS4A6 44345146 Ki = 3000 nM T95399 CY8L5Q 44354084 IC50 = 647 nM T95399 CVY98H 44354099 IC50 = 109 nM T95399 C0C2IS 44354283 IC50 = 12300 nM T95399 CX7TL1 44354301 IC50 = 29 nM T95399 CE65JT 44354322 IC50 = 167 nM T95399 CINT36 44354348 IC50 = 468 nM T95399 C8UCM7 44354349 IC50 = 200 nM T95399 CNR06G 44354350 IC50 = 181 nM T95399 CT43DB 44354362 IC50 = 844 nM T95399 C1EIY4 44354370 IC50 = 110 nM T95399 CHGM26 44354391 IC50 = 9 nM T95399 CI03FC 44354408 IC50 = 1860 nM T95399 CRXN57 44354446 IC50 = 25 nM T95399 CDE41K 44354454 IC50 = 80 nM T95399 CQ9IP7 44354455 IC50 = 57 nM T95399 CHTI61 44354456 IC50 = 140 nM T95399 CS7CE9 44354829 IC50 = 12 nM T95399 CIQM91 44354843 IC50 = 3 nM T95399 CU60QX 44354844 IC50 = 12 nM T95399 C4OX0H 44357872 IC50 = 98 nM T95399 CE36PI 44357873 IC50 = 89 nM T95399 C6UIG5 44357874 IC50 = 73 nM T95399 C7B6LO 44357907 IC50 = 56 nM T95399 CSEP-56 44357919 IC50 = 105 nM T95399 CS2VR8 44357925 IC50 = 83 nM T95399 CV4CE2 44357926 IC50 = 39 nM T95399 CZ3LM4 44357933 IC50 = 240 nM T95399 CTCI46 44357937 IC50 = 57 nM T95399 CS20RO 44357938 IC50 = 58 nM T95399 C3ZR9I 44358037 IC50 > 20000 nM T95399 C85KUT 44358038 IC50 = 550 nM T95399 CGEX65 44358070 IC50 = 2700 nM T95399 C6WE2Q 44358094 IC50 = 110 nM T95399 C8JV9Q 44358107 IC50 = 1700 nM T95399 CE3PV5 44358108 IC50 = 850 nM T95399 C6KXF8 44358150 IC50 = 2100 nM T95399 CBJ6P0 44358151 IC50 = 88 nM T95399 C20AUQ 44358152 IC50 > 20000 nM T95399 C3YGV2 44358155 IC50 = 69 nM T95399 C8EFT0 44358159 IC50 = 2440 nM T95399 CQ4RA3 44358172 IC50 > 20000 nM T95399 CGK1A5 44358173 IC50 = 6800 nM T95399 CTPE57 44358204 IC50 = 55 nM T95399 C3EW8Q 44358205 IC50 > 20000 nM T95399 CAK56U 44358343 IC50 = 2310 nM T95399 C65TFS 44358344 IC50 = 21700 nM T95399 CU7OF1 44358402 IC50 = 120 nM T95399 CT6J1N 44403045 IC50 = 2500 nM T95399 C9B7FV 44403049 IC50 = 5000 nM T95399 CT7JL5 44403050 IC50 > 10000 nM T95399 CT31XP 44403051 IC50 = 2500 nM T95399 CL6T2G 44403054 IC50 > 10000 nM T95399 C01GJK 44403058 IC50 = 480 nM T95399 C51UIK 44403142 IC50 > 10000 nM T95399 C6V2QU 44403153 IC50 = 160 nM T95399 CY03FE 44403159 IC50 > 10000 nM T95399 C12BMA 44403167 IC50 = 5700 nM T95399 C1Q0HV 44403170 IC50 = 710 nM T95399 C2FBL6 44403171 IC50 = 580 nM T95399 CG06DV 46905967 IC50 > 10000 nM T95399 CE94YF 52946782 Ki = 4600 nM T95399 CE41UW 56603813 Ki = 1020 nM T95399 C01YUK 56603814 Ki = 3270 nM T95399 C8N0LT 56603815 Ki = 1940 nM T95399 CD0U1K 57519731 IC50 = 291400 nM T95399 CS8NM0 118719323 Ki = 4200 nM T95399 D01BZE 73659 IC50 = 28000 nM T95399 D0E4SM 657140 IC50 = 900 nM T95399 D0F9RO 6918774 IC50 = 20000 nM T95399 D0S0AN 444746 IC50 = 500 nM T30495 D0E3TC 44259 IC50 = 0.37 nM T30495 C3VRO9 44557921 IC50 > 10000 nM T30495 CV63UL 67240318 IC50 > 10000 nM T30495 C1V3NZ 73425588 IC50 = 5.75 nM T30495 CYHR27 91664373 IC50 = 9 nM T30495 CL0YO5 118443595 IC50 > 100 nM T30495 CPHG43 135567142 IC50 = 4 nM T30495 C2MD1Q 155513187 IC50 > 10000 nM T21123 D0C9PZ 91754484 IC50 = 12 nM T21123 D0NU8J 117947097 IC50 = 9 nM T21123 CJB0A4 122826 EC50 > 100000 nM T21123 C37TUW 122838 EC50 > 100000 nM T21123 CJ5D7A 1278684 IC50 = 248 nM T21123 CV9RT4 1278687 IC50 > 30000 nM T21123 C2EL7S 6438762 EC50 = 2700 nM T21123 C1E7NA 9817550 EC50 = 700 nM T21123 C2ORD8 10316977 EC50 = 14800 nM T21123 CHQ84E 21589810 EC50 = 1200 nM T21123 C4NE0D 23245942 EC50 > 100000 nM T21123 CEYL14 23425818 EC50 = 4200 nM T21123 C14TIV 44566893 EC50 > 100000 nM T21123 CLW9G7 54584323 EC50 = 148900 nM T21123 CTJN02 54585297 EC50 = 183300 nM T21123 CXS1Z7 54585298 EC50 = 3400 nM T21123 C4Y7IG 54585299 EC50 = 11800 nM T21123 C6A2YK 54586240 EC50 = 107500 nM T21123 C3I1KH 54586242 EC50 = 6200 nM T21123 CF71NT 70697712 IC50 = 490 nM T21123 CAR63O 71457117 EC50 = 8700 nM T21123 CKN7X5 91663289 IC50 < 5 nM T21123 CUQ1W0 91810395 IC50 < 5 nM T21123 COR0A3 117942095 IC50 = 44400 nM T21123 CD7JT9 117942268 IC50 = 4400 nM T21123 C3UWY7 117942336 EC50 = 3700 nM T21123 CA5GJ3 117942346 IC50 = 4200 nM T21123 C5A0TS 117942380 IC50 < 5 nM T21123 C0WX5M 117942393 IC50 = 18200 nM T21123 CJK1C2 117942479 IC50 = 1200 nM T21123 CA07EP 117942585 IC50 = 52900 nM T21123 CTO03V 117942611 IC50 = 700 nM T21123 CZ65WM 117942644 IC50 = 180 nM T21123 C5Y1RM 117942651 IC50 = 31 nM T21123 C7SNI3 117942804 EC50 = 380 nM T21123 C1OHI0 117943024 IC50 = 22600 nM T21123 C3ZQK9 117943030 IC50 = 140 nM T21123 CVJD16 117947014 EC50 = 37 nM T21123 CRU39H 117947043 IC50 = 350 nM T21123 CVC19A 117947045 EC50 = 1900 nM T21123 CT64IZ 117947049 IC50 < 5 nM T21123 CS78OR 117947053 IC50 = 3600 nM T21123 CJ8TA1 117947087 IC50 = 10 nM T21123 CPZ9Y2 117947092 EC50 < 5 nM T21123 CUB2K7 117947096 EC50 = 4 nM T21123 CUX8M3 117947100 EC50 = 460 nM T21123 CN91AR 117947111 IC50 = 6500 nM T21123 CNDU29 117947115 EC50 = 930 nM T21123 CGMZ04 117947117 IC50 < 5 nM T21123 C23ZWM 117947131 IC50 = 34 nM T21123 CJ05VB 117947141 EC50 = 39 nM T21123 CJF37Q 118164921 EC50 = 13 nM T21123 CDV6W0 118165056 IC50 = 20 nM T21123 CGPW35 118165096 IC50 < 5 nM T21123 CI0WK9 118165112 EC50 = 7200 nM T21123 CKE42L 118183634 IC50 = 350 nM T21123 C4BFY8 118183648 IC50 < 5 nM T21123 CD6B3J 118183653 IC50 = 1100 nM T21123 CLC82K 118183703 EC50 = 9200 nM T21123 C2Z3IW 118183706 EC50 = 180 nM T21123 C4E6FD 118183707 EC50 = 32 nM T21123 CWL37Z 118183715 IC50 = 19600 nM T21123 C4IH0V 118183718 IC50 = 20 nM T21123 C3OS9F 118183719 IC50 < 5 nM T21123 C6J1KC 118183808 IC50 = 1700 nM T21123 CZ4M2R 121269926 IC50 = 3200 nM T21123 CV6KP1 121269947 IC50 < 5 nM T21123 CL9P4S 122506316 IC50 = 55 nM T21123 CTP7J6 122506359 EC50 = 240 nM T21123 C7VM2H 122506385 IC50 > 10000 nM T21123 CHN3O2 122506390 EC50 = 2900 nM T21123 CSV0Q5 134821994 IC50 < 5 nM T21123 CMJ23G 136075559 IC50 = 112 nM T21123 CV39WX 136268869 IC50 = 43 nM T21123 CGFU84 136268871 IC50 = 195 nM T21123 CN5SJ1 136268872 IC50 = 314 nM T21123 CPY3M7 136268873 IC50 = 97 nM T21123 C49QMW 136268879 IC50 = 87 nM T21123 CM4O5B 136268880 IC50 = 32 nM T21123 CK96MF 137036807 IC50 = 1000 nM T21123 CCFS85 137036808 IC50 > 30000 nM T21123 C1BME9 137036809 IC50 = 28300 nM T21123 C75PZK 137036810 IC50 > 30000 nM T21123 C5J3RC 137036811 IC50 > 30000 nM T21123 C85EID 137036812 IC50 = 108 nM T21123 C07MVZ 137036813 IC50 > 30000 nM T21123 C8XLD3 137036814 IC50 > 30000 nM T21123 C8MNO6 137036815 IC50 = 22300 nM T21123 CJK2M1 137036816 IC50 > 30000 nM T21123 C9USP2 137036817 IC50 > 30000 nM T21123 CJQK67 145952394 IC50 = 280 nM T21123 CJM8K0 145952445 IC50 = 280 nM T21123 CBVJ54 145953874 IC50 = 32 nM T21123 C4JC1V 145958339 IC50 = 12700 nM T21123 CAY73K 145960097 IC50 > 100000 nM T21123 CB72GT 145960173 IC50 = 4200 nM T21123 CPD5Z8 145971957 IC50 = 16 nM T09133 D09XZL 56962369 IC50 = 7.5 nM T09133 D0E3TC 44259 IC50 = 102 nM T09133 CDN96Q 4789349 IC50 = 95 nM T09133 C1X6VQ 11589985 IC50 = 64 nM T09133 CE97MA 17646732 IC50 = 2320 nM T09133 C8I6DU 24408249 IC50 = 24100 nM T09133 C7TK2M 25185020 IC50 = 1.1 nM T09133 C0MK3N 25185023 IC50 = 1.9 nM T09133 CYZ7N3 25186125 IC50 = 2.9 nM T09133 C5O3PU 25186126 IC50 = 1.7 nM T09133 C0SJ9Y 25186127 IC50 = 1.2 nM T09133 CN51GJ 25187230 IC50 = 37 nM T09133 C0O2LX 25187232 IC50 = 3.9 nM T09133 C8U4GS 25187234 IC50 = 2.3 nM T09133 C1VD2L 25187799 IC50 = 5.5 nM T09133 CW90ZX 25187801 IC50 = 3 nM T09133 CKLS38 25187803 IC50 = 2.7 nM T09133 CK91LH 25348412 IC50 = 120 nM T09133 CXQ04O 25348413 IC50 = 110 nM T09133 C0LHA7 26534648 IC50 = 3200 nM T09133 C3T6AM 26555947 IC50 = 53 nM T09133 CC71QJ 27666048 IC50 = 39 nM T09133 CZ5X3K 27666050 IC50 = 52 nM T09133 CD71LI 27666053 IC50 = 81 nM T09133 C0HPA6 27666060 IC50 = 120 nM T09133 CNLG15 37311853 IC50 = 3 nM T09133 C23UAJ 44481840 IC50 = 2.7 nM T09133 CQML65 44482388 IC50 = 1.9 nM T09133 C6PZQ2 44542470 IC50 = 4.2 nM T09133 CTW70K 44542471 IC50 = 133 nM T09133 C7RUS4 44542472 IC50 = 76 nM T09133 CBG9C0 44542473 IC50 = 650 nM T09133 CR10TV 44542474 IC50 = 1500 nM T09133 CH2S9Y 44542475 IC50 = 300 nM T09133 CY93VX 44542622 IC50 = 140 nM T09133 C1X6MO 44542623 IC50 = 800 nM T09133 C68ABN 44542624 IC50 = 11500 nM T09133 CPB70M 44542625 IC50 = 1300 nM T09133 CAK4P7 44542626 IC50 = 520 nM T09133 CO28NP 44542627 IC50 = 92 nM T09133 CKJ9F7 44542628 IC50 = 38 nM T09133 CT6V9L 44542772 IC50 = 11 nM T09133 CG8P4D 44542773 IC50 = 3.9 nM T09133 CJOT19 44542774 IC50 = 16 nM T09133 CWVM19 44542775 IC50 = 8.1 nM T09133 CD5C7M 44542776 IC50 = 1.2 nM T09133 C6DJZ1 44542921 IC50 = 4.2 nM T09133 C4KTM9 44542922 IC50 > 1000 nM T09133 CCDQ50 44542923 IC50 = 6.8 nM T09133 CAY0M1 44542924 IC50 = 1.6 nM T09133 C64VZL 44542925 IC50 = 1.8 nM T09133 CRZ79W 44542926 IC50 = 1.5 nM T09133 CE0O4B 44543079 IC50 = 3.2 nM T09133 CQT48I 44543080 IC50 = 1.2 nM T09133 CDI73J 44543081 IC50 = 3.5 nM T09133 CF2WJ9 44543083 IC50 = 3 nM T09133 C9CP0U 44543084 IC50 = 3.4 nM T09133 C3VRO9 44557921 IC50 > 10000 nM T09133 C35PRM 46584923 IC50 = 1000 nM T09133 CV0CZ5 52942728 IC50 = 362 nM T09133 CIVE91 52949671 IC50 = 3.05 nM T09133 C7LAS5 56965901 IC50 = 85 nM T09133 C1XZ2W 57920198 IC50 = 4.8 nM T09133 CN23UC 57920200 IC50 = 3.2 nM T09133 C7CGB9 57920201 IC50 = 5.1 nM T09133 C5ROV3 57920202 IC50 = 138 nM T09133 CO7SX4 57920205 IC50 < 1 nM T09133 C9PKH2 57920206 IC50 = 1 nM T09133 C3V6MX 57920210 IC50 = 7.3 nM T09133 C86YRV 58688296 IC50 = 382 nM T09133 C8AT5N 58688313 IC50 = 28 nM T09133 C09YWX 58688317 IC50 = 245 nM T09133 C4Q2HL 58688342 IC50 = 202 nM T09133 C0LK4S 58688380 IC50 = 12 nM T09133 CNVK41 58688409 IC50 = 1531 nM T09133 CJI0Q4 58688436 IC50 = 50000 nM T09133 CK1AO4 58688444 IC50 = 16 nM T09133 CZ0J6F 58688467 IC50 = 1232 nM T09133 CPE98M 58688474 IC50 = 50000 nM T09133 CDOK25 58688484 IC50 = 1545 nM T09133 CHO5G0 58688561 IC50 = 141 nM T09133 CP2JK1 58688569 IC50 = 311 nM T09133 CIV53P 58688575 IC50 = 16 nM T09133 C2T8UL 58688642 IC50 = 1222 nM T09133 C3IZ0N 66548972 IC50 = 164 nM T09133 CKW80R 66549342 IC50 = 157 nM T09133 CENC12 66549526 IC50 = 103 nM T09133 C13EIQ 66549529 IC50 = 273 nM T09133 CV63UL 67240318 IC50 > 10000 nM T09133 CIJ5L9 70682556 IC50 = 810 nM T09133 C9IB8C 70684645 IC50 = 59 nM T09133 CH08ZN 70690951 IC50 = 171 nM T09133 CK0CH3 70697188 IC50 = 760 nM T09133 CH5QO0 70812854 IC50 = 90 nM T09133 CGS60U 70812857 IC50 = 133 nM T09133 C1E6PA 91938057 IC50 = 0.7 nM T09133 C8N9TC 109060734 IC50 = 22 nM T09133 CX0UO9 109060735 IC50 = 22 nM T09133 CTLS12 117918919 IC50 = 48 nM T09133 CH4GF2 117918922 IC50 = 3 nM T09133 C1MF8V 118720892 IC50 = 51 nM T09133 C2SKL7 118720893 IC50 = 540 nM T09133 C57RIT 118720894 IC50 > 27000 nM T09133 CP0M9J 118720895 IC50 > 27000 nM T09133 CEX7M3 118720896 IC50 = 34 nM T09133 C3OQ6B 118720897 IC50 = 19 nM T09133 C5ZHM6 118720898 IC50 = 92 nM T09133 C67CBN 118720899 IC50 = 1640 nM T09133 CY9LH1 118720900 IC50 = 900 nM T09133 C5M9IY 118720901 IC50 = 36 nM T09133 C4RS8L 118720902 IC50 > 27000 nM T09133 C9RH4M 118720903 IC50 > 27000 nM T09133 COZ78F 118720904 IC50 > 27000 nM T09133 CQ72EV 118720905 IC50 = 19 nM T09133 CRD40E 118720906 IC50 = 52 nM T09133 C5K0FW 118720907 IC50 = 160 nM T09133 CBIC45 118720908 IC50 = 1200 nM T09133 C9NV2Q 118720909 IC50 = 1500 nM T09133 C7RG0Y 118720910 IC50 = 1530 nM T09133 C6KSE8 118720911 IC50 > 27000 nM T09133 CDI09N 118720912 IC50 = 22 nM T09133 C8M5BH 118720913 IC50 = 100 nM T09133 CGWD43 118720914 IC50 = 90 nM T09133 C5J0IM 118721274 IC50 = 1.2 nM T09133 CIV07K 118721275 IC50 = 660 nM T09133 C3TFZ5 118721276 IC50 = 9.9 nM T09133 CUF3R4 118721277 IC50 = 180 nM T09133 C6OTL0 118721279 IC50 = 220 nM T09133 C2G6BA 118721535 IC50 = 26 nM T09133 C7LD6O 118721536 IC50 > 1000 nM T09133 C5BHU3 118721537 IC50 = 330 nM T09133 CE1N0X 118721538 IC50 = 210 nM T09133 C29CGB 118721539 IC50 = 110 nM T09133 CM1E6U 118721540 IC50 = 2.2 nM T09133 C1ACJ0 122189152 IC50 < 1 nM T09133 CTOX13 122189153 IC50 = 1.5 nM T09133 CA0NQ6 122189154 IC50 = 7.4 nM T09133 CXK73S 122189155 IC50 = 12 nM T09133 CUYA85 122189156 IC50 < 1 nM T09133 CQS34F 122189157 IC50 < 1 nM T09133 CE13UV 122189158 IC50 = 7.7 nM T09133 C4E8IF 122189159 IC50 = 2.1 nM T09133 CCT83H 122189160 IC50 = 2.2 nM T09133 CY23RV 122189161 IC50 = 4.6 nM T09133 CFJR29 122189162 IC50 < 1 nM T09133 CEX47Y 122189163 IC50 = 13 nM T09133 CUB9Q5 122189164 IC50 = 193 nM T09133 C63OQZ 122189165 IC50 = 274 nM T09133 CG51VB 122189166 IC50 = 1860 nM T09133 CH74JB 122189167 IC50 = 9.6 nM T09133 C0SO5F 122189168 IC50 > 10000 nM T09133 CUML53 122189169 IC50 = 4560 nM T09133 C23PWJ 122189170 IC50 > 10000 nM T09133 C4M6BZ 122189171 IC50 = 494 nM T09133 C5ZO6J 122189172 IC50 > 10000 nM T09133 C36LON 122189173 IC50 = 4 nM T09133 C5IDL1 122189174 IC50 = 2.8 nM T09133 CTQ9U7 122189175 IC50 = 8 nM T09133 C31YGS 122189176 IC50 = 1.6 nM T09133 CC48FJ 122189177 IC50 = 1.4 nM T09133 CV2U0H 122192497 IC50 = 1 nM T09133 C9EA4L 127045691 IC50 = 32 nM T09133 C6HL1A 127045692 IC50 = 2 nM T09133 CFH0O6 127045693 IC50 = 4.8 nM T09133 CHY13L 127045694 IC50 = 11 nM T09133 CM6X8C 127045695 IC50 = 62 nM T09133 C5SGK1 127045876 IC50 = 0.3 nM T09133 CF52WT 127045877 IC50 = 0.3 nM T09133 C1R3KZ 127045878 IC50 < 0.1 nM T09133 CBH61K 127045879 IC50 < 0.1 nM T09133 C0A8UZ 127045880 IC50 = 0.9 nM T09133 CXY8M4 127046486 IC50 = 17 nM T09133 CF17NZ 127046673 IC50 = 27 nM T09133 C8ZC9B 127046674 IC50 = 122 nM T09133 C6ID3B 127046675 IC50 = 41 nM T09133 C0T9LZ 127046676 IC50 = 22 nM T09133 CD98AI 127046677 IC50 = 7.1 nM T09133 CL9YK2 127046847 IC50 < 0.1 nM T09133 CQB3G8 127046988 IC50 = 1.4 nM T09133 CY2N5R 127046989 IC50 < 0.1 nM T09133 CU94AT 127046990 IC50 = 0.2 nM T09133 C68KQH 127046991 IC50 < 0.1 nM T09133 CF8OZ9 127047123 IC50 = 0.2 nM T09133 CZ7CJ6 127047267 IC50 = 0.2 nM T09133 CLX36O 127047268 IC50 = 4.5 nM T09133 CL27TP 127047269 IC50 = 12 nM T09133 CAF53U 127047270 IC50 = 3.7 nM T09133 CI3J6M 127047397 IC50 = 105 nM T09133 CISD39 127047398 IC50 = 700 nM T09133 C14ELG 127047544 IC50 < 0.1 nM T09133 CMU47C 127047575 IC50 = 0.7 nM T09133 CLJ98V 127047576 IC50 = 0.1 nM T09133 CL5X2G 127047577 IC50 < 0.1 nM T09133 CTU50H 127047686 IC50 = 0.1 nM T09133 CEC5V6 127047687 IC50 = 0.9 nM T09133 C8T9RS 127047688 IC50 = 0.4 nM T09133 C1YHM5 127047689 IC50 = 23 nM T09133 CB8G2L 127047708 IC50 = 13 nM T09133 CIBT73 127047709 IC50 = 0.8 nM T09133 C4G0YA 127047710 IC50 = 0.4 nM T09133 CD06GZ 127047823 IC50 = 12 nM T09133 C2NQF1 127047824 IC50 = 0.4 nM T09133 CAW6X5 127047919 IC50 = 1.4 nM T09133 C3YE1D 127048049 IC50 = 1 nM T09133 C2QP4D 127048050 IC50 = 0.2 nM T09133 C2JF4I 127048078 IC50 = 31 nM T09133 C3B4HT 136003186 IC50 > 12500 nM T09133 C6VB3O 145925651 IC50 >= 5000 nM T09133 C2MD1Q 155513187 IC50 = 46 nM T09133 D07XWC 44477445 IC50 = 0.9 nM T09133 D0F6NZ 58688690 IC50 = 173 nM T09133 D0FC4Y 46192505 IC50 = 38 nM T09133 D0S0XD 58688563 IC50 = 8 nM T09133 D0YI1Z 44543082 IC50 = 0.8 nM T60857 D05FTJ 4044 Ki = 300 nM T60857 D06YPU 39912 IC50 = 32700 nM T60857 D08IFL 4037 IC50 = 540 nM T60857 D0A1PX 3394 IC50 = 1560 nM T60857 D0B2WJ 3371 IC50 = 410 nM T60857 D0DJ1B 156391 IC50 = 180 nM T60857 D0R1QE 3672 IC50 = 10000 nM T60857 D0R1RS 3715 IC50 = 100 nM T60857 D0W8WB 2353 IC50 = 5900 nM T60857 D0H7XJ 25210792 IC50 = 120 nM T60857 D0E2TY 71523527 IC50 = 340 nM T60857 D0F0PK 4711697 IC50 = 960 nM T60857 D0G8VB 66706413 Ki = 31 nM T60857 D0GY2Z 11394647 IC50 = 220 nM T60857 D0M6LX 56851703 IC50 = 80 nM T60857 C59UQE 6279 IC50 = 2511.89 nM T60857 C8Z0TY 6813 IC50 = 70000 nM T60857 CQP80E 15339 IC50 = 5670 nM T60857 CHM42L 18464 Ki = 23000 nM T60857 C0EX5S 22630 IC50 = 3560 nM T60857 CQ50AX 32176 IC50 = 650 nM T60857 C68GPN 66563 IC50 = 44000 nM T60857 CBNY48 69146 IC50 = 180000 nM T60857 CNWC30 76151 IC50 > 100000 nM T60857 COF34W 83293 IC50 = 150 nM T60857 C0BE1A 85472 IC50 = 240 nM T60857 CE6G3T 97298 IC50 = 980 nM T60857 CYOP05 101403 IC50 = 40 nM T60857 CFG89D 119702 IC50 = 570 nM T60857 CZS90Q 119703 IC50 = 140 nM T60857 C40FKV 152155 IC50 = 360 nM T60857 C6A0PT 169118 IC50 = 50 nM T60857 C0X8NW 176925 IC50 = 100 nM T60857 CE1DI3 201986 IC50 = 160 nM T60857 CV4YO6 202774 IC50 = 2220 nM T60857 C4U5MD 202918 IC50 = 90 nM T60857 C83PSY 205081 IC50 = 40 nM T60857 CHU43L 205082 IC50 = 2740 nM T60857 CDZ9Q2 256062 IC50 = 39000 nM T60857 C2J8XS 259483 IC50 > 30000 nM T60857 C7Y5GE 285710 Ki = 111000 nM T60857 C1RFC8 292331 IC50 = 2790 nM T60857 CN12SD 313797 IC50 = 1320 nM T60857 CY4D0W 344658 IC50 = 7220 nM T60857 C4SM3C 362740 Ki = 148000 nM T60857 CFA40G 368710 Ki = 2730 nM T60857 CP4ZX0 459316 IC50 = 70 nM T60857 CG8W5M 527316 IC50 = 7590 nM T60857 C9NB2A 579839 Ki = 82000 nM T60857 CN29IX 591357 Ki = 72000 nM T60857 C8Y7MQ 610479 Ki = 8 nM T60857 CM0KQ2 614334 IC50 = 30 nM T60857 C6H0SZ 651438 IC50 = 47 nM T60857 C90SBI 652676 IC50 = 16500 nM T60857 CZX57W 668656 Ki = 76000 nM T60857 CK98GL 673729 Ki = 54000 nM T60857 CPY40J 682194 Ki = 4000 nM T60857 CNX4A8 703764 Ki = 118000 nM T60857 C0MI2B 712934 IC50 = 13 nM T60857 CLD28R 737166 IC50 > 30000 nM T60857 C51SXE 745875 IC50 > 30000 nM T60857 C8C3KO 745878 IC50 = 140 nM T60857 CKB04T 747663 IC50 = 24200 nM T60857 CK92FW 754983 IC50 = 350 nM T60857 CYC81A 767169 Ki = 44000 nM T60857 CB8MG7 791238 IC50 = 20300 nM T60857 C7QGF8 794747 Ki = 12000 nM T60857 CAM37G 794776 Ki = 36000 nM T60857 C64FJR 804306 Ki = 148000 nM T60857 C6ZK4Y 838922 IC50 = 500 nM T60857 CC8Q9P 851812 IC50 > 30000 nM T60857 CBZ73S 863775 IC50 > 1000 nM T60857 C4MGO9 878243 IC50 = 6100 nM T60857 CKY1S3 946901 IC50 = 5300 nM T60857 C94NFJ 976980 IC50 = 110 nM T60857 CF7D8A 977233 IC50 = 3800 nM T60857 CPS8Z9 1081072 Ki = 142000 nM T60857 C7S6UP 1217101 IC50 = 13 nM T60857 CI9QB4 2315499 IC50 = 199.53 nM T60857 CRU7Q2 2473940 IC50 = 218.78 nM T60857 CU21OR 2712225 IC50 = 13 nM T60857 CHB74O 2832029 Ki = 87000 nM T60857 CA29GS 2865352 IC50 > 25000 nM T60857 CU5N7J 2886767 IC50 > 30000 nM T60857 C2QB1O 2925862 IC50 = 15200 nM T60857 CP6OX3 3136316 IC50 = 570 nM T60857 C8TDV1 3139647 IC50 = 6730 nM T60857 CZEC70 3292097 IC50 = 160 nM T60857 CO0S9F 3493153 IC50 = 227 nM T60857 CT3Y0G 3626723 IC50 = 12600 nM T60857 COL1U7 3706434 IC50 > 30000 nM T60857 CH0GV6 3807505 IC50 = 208.93 nM T60857 CM2Q7U 3897551 IC50 = 533 nM T60857 CP63TL 4342938 IC50 = 3960 nM T60857 CK4XO2 4393667 IC50 > 25000 nM T60857 CKZ83R 4416918 IC50 > 30000 nM T60857 C14IYN 4549649 IC50 > 30000 nM T60857 C0U2VG 4712246 IC50 = 2370 nM T60857 CAKX74 4763851 IC50 = 30 nM T60857 C4JQ5B 4763963 IC50 = 30 nM T60857 CNPV35 5018304 IC50 = 2600 nM T60857 C3NRJ7 5281166 Ki = 24000 nM T60857 CRXZ63 5281929 Ki = 153000 nM T60857 CJY35S 5315107 IC50 = 121100 nM T60857 CSG8D7 6440361 IC50 = 15000 nM T60857 CAN3U5 6612512 IC50 = 460 nM T60857 CQHW10 7063081 IC50 = 398.11 nM T60857 CB5TF7 7063083 IC50 = 31.62 nM T60857 CSOQ75 8404968 IC50 > 30000 nM T60857 C7JU0L 9947201 Ki = 46 nM T60857 CW29AN 10106489 IC50 = 5190 nM T60857 CZQU30 11184397 IC50 = 54 nM T60857 CW18VN 11186887 IC50 = 710 nM T60857 C6XH3D 11187310 IC50 = 140 nM T60857 CQ4U8H 11187365 IC50 = 42 nM T60857 CBEO86 11256258 IC50 = 49 nM T60857 C9J2TX 11276572 IC50 = 2210 nM T60857 CE4M5J 11345534 IC50 = 1190 nM T60857 C2X1TU 11350052 IC50 = 72 nM T60857 CW5S0P 11357272 IC50 = 2500 nM T60857 CSOI34 11371225 IC50 = 20 nM T60857 CXDE57 11393656 IC50 = 66 nM T60857 C8QTI1 11416926 IC50 = 16 nM T60857 C5V3UY 11417322 IC50 = 28 nM T60857 C14YIN 11425050 IC50 = 490 nM T60857 C5RP9Y 11450564 IC50 = 160 nM T60857 C7TZ6Q 11470189 IC50 = 1670 nM T60857 C9PYZ6 11473705 IC50 = 19 nM T60857 CP45FG 11474483 IC50 = 107 nM T60857 CB1KD0 11623967 IC50 > 30000 nM T60857 CFQ0M2 11637363 IC50 = 1200 nM T60857 CAYU53 11987804 IC50 = 3.2 nM T60857 CY4L5J 12648027 IC50 = 1660 nM T60857 C9LN3B 12658319 IC50 = 2240 nM T60857 C61PIM 12658320 IC50 = 740 nM T60857 CO93UK 12847796 IC50 = 130 nM T60857 CRI5B0 12850341 IC50 = 940 nM T60857 CX26MU 13098689 IC50 > 30000 nM T60857 C4RIQ8 13105472 IC50 = 320 nM T60857 CK4R8I 13105473 IC50 = 500 nM T60857 CRK0V1 13292509 IC50 = 120 nM T60857 C1TCI4 13521073 IC50 = 2530 nM T60857 C3JP4Q 14380427 IC50 = 890 nM T60857 C1WJ2D 16070041 IC50 > 50000 nM T60857 C2K8UZ 16738708 IC50 = 67.61 nM T60857 CBH78X 16771604 IC50 = 310 nM T60857 CWYV84 16775967 IC50 = 2900 nM T60857 C34NRV 16776644 IC50 = 840 nM T60857 C3IS5U 16778344 IC50 = 34 nM T60857 CQVJ02 16876789 Ki = 144000 nM T60857 CHZ06B 17217372 IC50 = 12500 nM T60857 CNBH53 17217648 IC50 = 5940 nM T60857 CTA0Z9 18096680 IC50 = 24 nM T60857 C6QW7Z 18096684 IC50 > 30000 nM T60857 C8U0MV 19585911 Ki = 117000 nM T60857 CRF3A4 19614435 IC50 = 200 nM T60857 C2SUP9 19614516 IC50 = 15 nM T60857 C2XTZ6 19749436 IC50 = 800 nM T60857 C1Z5JY 19749467 IC50 = 640 nM T60857 CR6KB3 19849814 IC50 = 270 nM T60857 C8NV4Z 19849815 IC50 = 2440 nM T60857 CXNC35 20334995 IC50 = 100 nM T60857 C8KNB1 20335074 IC50 = 120 nM T60857 CT5NS8 20335119 IC50 = 60 nM T60857 CBST06 20486899 IC50 = 1050 nM T60857 C58WUL 20937276 IC50 = 11 nM T60857 CK1XQ5 21548774 IC50 = 160 nM T60857 CJ4KW0 21737210 IC50 = 2650 nM T60857 CDM3I1 21747812 IC50 = 380 nM T60857 CW8ZL7 21819689 IC50 = 340 nM T60857 C1V4IN 22142202 IC50 > 30000 nM T60857 C1MB9W 22564610 IC50 = 1890 nM T60857 CDG65Y 22607959 Ki = 21000 nM T60857 CPV67M 23456902 IC50 = 1090 nM T60857 CTQM87 25210756 IC50 = 0.34 nM T60857 C8YKC6 25210766 IC50 = 2.1 nM T60857 C4FO5I 25269617 IC50 = 6.1 nM T60857 C53PAL 25269954 IC50 = 10 nM T60857 CJBG70 25269955 IC50 = 2.9 nM T60857 C8R2PD 25755895 IC50 = 602.56 nM T60857 C8GK5A 27678343 IC50 = 14 nM T60857 C3OEC9 31673322 IC50 > 30000 nM T60857 CZQ27X 34680232 IC50 = 480 nM T60857 CU24HX 38274995 IC50 = 31 nM T60857 C1KEM3 42346590 IC50 = 22 nM T60857 C8J1AG 43238244 IC50 = 150 nM T60857 C5KA7X 43358888 IC50 = 2060 nM T60857 C8DQ4J 43358934 IC50 = 40 nM T60857 C3A7JX 43421689 IC50 = 230 nM T60857 CBPV58 43461651 IC50 = 4210 nM T60857 CJN73T 43461652 IC50 = 290 nM T60857 CCFP75 44141469 IC50 = 169.82 nM T60857 CA2O1E 44451451 IC50 = 139200 nM T60857 C5KMP1 44576210 IC50 = 9.5 nM T60857 CAN59E 45035007 IC50 = 14800 nM T60857 C9S8MO 45414370 IC50 = 1440 nM T60857 C4BL6F 45414688 IC50 = 140 nM T60857 CMXG67 45415196 IC50 = 330 nM T60857 CWC8L0 45415334 IC50 = 208.93 nM T60857 C47DTG 45732904 IC50 > 30000 nM T60857 C6GK7O 46213655 IC50 = 10700 nM T60857 CZ29QD 46861569 IC50 = 70 nM T60857 CQ9SI3 46909652 IC50 = 140 nM T60857 CU7ST1 51346826 IC50 = 60 nM T60857 CJP9O3 51346855 IC50 = 10600 nM T60857 C1OJ0M 53316888 IC50 = 120 nM T60857 CG79XF 53316889 IC50 = 280 nM T60857 C08TYZ 53317604 IC50 = 17600 nM T60857 C7RFD6 53323514 IC50 = 700 nM T60857 CRXD98 53324830 IC50 = 130 nM T60857 CM1L7E 53326266 IC50 = 69800 nM T60857 CN48MT 53326634 IC50 = 8600 nM T60857 CU5O2P 54159801 IC50 = 250 nM T60857 CZL92O 54436150 IC50 = 570 nM T60857 CKMN16 55049196 IC50 = 870 nM T60857 C4JXC1 55050538 IC50 = 3390 nM T60857 CLO87D 56964583 IC50 = 40 nM T60857 C7GR8D 57563309 IC50 = 11340 nM T60857 CX9P8K 57563344 IC50 = 130 nM T60857 CIZ81B 57819796 IC50 = 360 nM T60857 C1KA9P 57960521 IC50 = 12100 nM T60857 CBWL65 59512779 IC50 = 501.19 nM T60857 C6K5DO 59529913 IC50 = 33 nM T60857 CX97VG 59529919 IC50 = 12 nM T60857 C7ZY8I 59529925 IC50 = 2100 nM T60857 C6AP5R 59529928 IC50 = 4.5 nM T60857 C84XCR 59529932 IC50 = 37 nM T60857 CYN75V 59787536 IC50 = 7540 nM T60857 C3GT4B 60008666 IC50 = 1900 nM T60857 C6Z5MD 62230856 IC50 = 1180 nM T60857 C74APH 62231529 IC50 = 2530 nM T60857 C2AH6B 62313636 IC50 = 560 nM T60857 C3NV9G 63527647 IC50 = 930 nM T60857 CKX28S 64259878 IC50 > 30000 nM T60857 CCX5A7 66706325 IC50 = 120 nM T60857 C3DSO7 67474725 IC50 = 250 nM T60857 C23ZWP 68881866 IC50 = 13600 nM T60857 C9B5DN 70681846 IC50 = 1350 nM T60857 C35QMX 70681892 IC50 = 160 nM T60857 C2YG4K 70681893 IC50 = 500 nM T60857 CVAQ08 70683951 IC50 = 80 nM T60857 CL6N0V 70683952 IC50 = 690 nM T60857 CFI0L4 70683953 IC50 = 140 nM T60857 CM4P1O 70683954 IC50 = 1650 nM T60857 CD31CV 70683956 IC50 = 1880 nM T60857 CTZ15F 70683957 IC50 = 3570 nM T60857 CUNQ68 70686076 IC50 = 600 nM T60857 CTZ9Y6 70686077 IC50 = 610 nM T60857 C1OG6L 70686078 IC50 = 900 nM T60857 CXM5L3 70686079 IC50 = 1820 nM T60857 C7RL9Y 70686090 IC50 = 250 nM T60857 CAW04I 70686144 IC50 = 60 nM T60857 CC7L6S 70686145 IC50 = 150 nM T60857 C8XFE2 70686744 IC50 = 7500 nM T60857 C8YN0K 70688201 IC50 = 2220 nM T60857 CXBP89 70688202 IC50 = 1160 nM T60857 C1GQ2Z 70688203 IC50 = 2260 nM T60857 CO2HN4 70688204 IC50 = 1940 nM T60857 CICR62 70688205 IC50 = 1550 nM T60857 C8LKA9 70688206 IC50 = 1760 nM T60857 C1BLO2 70688208 IC50 = 610 nM T60857 C08ZYA 70688209 IC50 = 960 nM T60857 CVHY13 70688223 IC50 = 2910 nM T60857 CH90MN 70688224 IC50 = 1080 nM T60857 C3XPR8 70688285 IC50 = 220 nM T60857 CY7RT3 70690226 IC50 = 470 nM T60857 C1B0SE 70690227 IC50 = 250 nM T60857 C6Z0JO 70690228 IC50 = 280 nM T60857 CL4OA1 70690231 IC50 = 1650 nM T60857 CG50ZA 70690235 IC50 = 1640 nM T60857 CGPL20 70690246 IC50 > 30000 nM T60857 C71NSQ 70690294 IC50 = 1730 nM T60857 C2KS5G 70690295 IC50 = 1450 nM T60857 C6Q0LD 70692396 IC50 = 3060 nM T60857 CAD0Y1 70692398 IC50 = 650 nM T60857 C6TFC7 70692399 IC50 = 1170 nM T60857 C76ZQL 70692400 IC50 = 260 nM T60857 CPM0Z9 70692416 IC50 = 360 nM T60857 CFB31J 70694447 IC50 = 1730 nM T60857 CEDW62 70694448 IC50 = 1110 nM T60857 CQ5XH2 70694449 IC50 = 4440 nM T60857 CUM5H0 70694450 IC50 = 980 nM T60857 CWZ83L 70696515 IC50 = 730 nM T60857 CP37LD 70696516 IC50 = 560 nM T60857 C6K9WV 70696525 IC50 = 40 nM T60857 C2E6PC 70696565 IC50 = 80 nM T60857 CT7VJ2 70696566 IC50 = 500 nM T60857 CJ8DC4 70848211 IC50 = 160 nM T60857 CAQ8Y4 70848221 IC50 = 770 nM T60857 CLT07E 70848223 IC50 = 1100 nM T60857 CTV5N1 71449917 IC50 = 740 nM T60857 CB3S2M 71449918 IC50 = 24400 nM T60857 CC6P3X 71449919 IC50 = 14 nM T60857 C3LQO4 71449920 IC50 = 8.511 nM T60857 C76ZTD 71449921 IC50 = 10.96 nM T60857 CSZ1A6 71449925 IC50 = 390 nM T60857 C8U6ER 71451741 IC50 = 389.05 nM T60857 C48MFU 71451742 IC50 = 19.95 nM T60857 C3VMQ6 71451743 IC50 = 640 nM T60857 C10MJH 71451744 IC50 = 15.85 nM T60857 CIZ9J2 71451745 IC50 = 21.88 nM T60857 CER26G 71453564 IC50 = 35 nM T60857 CAY38B 71453565 IC50 > 30000 nM T60857 C8JXA5 71453566 IC50 = 29 nM T60857 CE0Y1Z 71453567 IC50 = 10.96 nM T60857 CEWP50 71453568 IC50 = 14 nM T60857 CIXZ83 71453569 IC50 = 17 nM T60857 C4K9SD 71453570 IC50 = 38.9 nM T60857 CBE86R 71453571 IC50 = 38 nM T60857 CJ6HT9 71455288 IC50 > 30000 nM T60857 CI4OM7 71455289 IC50 = 9.5 nM T60857 CX8MR1 71455290 IC50 = 891.25 nM T60857 CGI45B 71455291 IC50 = 68 nM T60857 CQFA31 71455292 IC50 = 12 nM T60857 CCMA45 71455293 IC50 = 42 nM T60857 CLSV31 71455294 IC50 = 24 nM T60857 CP9KX8 71455295 IC50 = 28.84 nM T60857 CP81EL 71455296 IC50 = 39 nM T60857 CHVS69 71455297 IC50 = 12 nM T60857 CK41AQ 71457072 IC50 = 550 nM T60857 CEKQ80 71457073 IC50 = 16.98 nM T60857 CJ58EM 71457074 IC50 = 26.92 nM T60857 CAZ0P5 71458926 IC50 = 61.66 nM T60857 CFGY71 71458927 IC50 = 28.84 nM T60857 CAB3N5 71458928 IC50 = 19 nM T60857 C8TR7X 71458929 IC50 = 218.78 nM T60857 C3QZE6 71458930 IC50 = 52.48 nM T60857 CF9Y4G 71458937 IC50 = 42 nM T60857 C3YJ4O 71460743 IC50 = 346.74 nM T60857 CQP51J 71460744 IC50 = 266 nM T60857 C6INL1 71460745 IC50 = 530 nM T60857 C2C0NS 71460748 IC50 = 12.88 nM T60857 CZ0AW1 71460749 IC50 = 1310 nM T60857 C5W7XO 71462462 IC50 > 30000 nM T60857 COG2J6 71462463 IC50 = 450 nM T60857 CWY04T 71462464 IC50 = 500 nM T60857 CHD29O 71462465 IC50 = 20.89 nM T60857 CGC6R1 71462466 IC50 = 740 nM T60857 COG3Y9 71462467 IC50 = 15.85 nM T60857 C6LCH7 71523525 IC50 = 500 nM T60857 CU3RF0 71523636 IC50 = 90 nM T60857 CPN8U4 71550737 IC50 = 210 nM T60857 CP86IK 71600419 IC50 = 12000 nM T60857 CJT9O7 71600420 IC50 = 12400 nM T60857 CQ2CF5 71600555 IC50 = 1190 nM T60857 C45ZRI 71600556 IC50 = 8820 nM T60857 CX9VP2 71600557 IC50 = 2070 nM T60857 C7PRA1 71600558 IC50 = 2650 nM T60857 CDN0R1 71600559 IC50 = 3730 nM T60857 CXND28 71600681 IC50 = 2090 nM T60857 CHE4U0 71600682 IC50 = 6340 nM T60857 CTZ2F6 71600683 IC50 = 5800 nM T60857 CD9JQ7 71600684 IC50 = 7860 nM T60857 C1XRD3 71600685 IC50 = 2520 nM T60857 CWB2S7 71600814 IC50 = 1110 nM T60857 CF0EW8 71600815 IC50 = 3970 nM T60857 C8IB2N 71600816 IC50 = 1940 nM T60857 CJZ0F7 71600817 IC50 = 120 nM T60857 C5MU9P 71600818 IC50 = 290 nM T60857 C49RBT 71600819 IC50 = 5530 nM T60857 CZ50CS 71600944 IC50 = 1440 nM T60857 CY0N3Z 71600945 IC50 = 3110 nM T60857 CU5K0V 71600946 IC50 = 2540 nM T60857 CW21EH 71600947 IC50 = 3250 nM T60857 CU75MD 71600948 IC50 = 1110 nM T60857 C82PCX 71601068 IC50 = 2500 nM T60857 CRJ60N 71601070 IC50 = 2650 nM T60857 CK1XQ4 71601071 IC50 = 4690 nM T60857 CYZC34 71601072 IC50 = 5070 nM T60857 CORM85 71653635 IC50 = 11880 nM T60857 CH72JT 71653636 IC50 = 19 nM T60857 CQ2OU4 71653778 IC50 = 8980 nM T60857 C03XEN 71653779 IC50 = 1550 nM T60857 C3K6MN 71653780 IC50 = 21200 nM T60857 CC6N5U 71653934 IC50 > 30000 nM T60857 CF02UQ 71653935 IC50 = 5610 nM T60857 CFY4W3 71653936 IC50 = 3770 nM T60857 C4BY7P 71653937 IC50 > 30000 nM T60857 CH4O8N 71653938 IC50 > 30000 nM T60857 CVL62B 71653939 IC50 = 10200 nM T60857 CP49BQ 71653940 IC50 > 30000 nM T60857 C8B6LQ 71653941 IC50 = 2770 nM T60857 CH6M2D 71654023 IC50 = 38700 nM T60857 CH36YF 71654026 IC50 = 86600 nM T60857 C2VL9B 71654027 IC50 = 10800 nM T60857 CQ57DL 71654028 IC50 = 17000 nM T60857 C5P8ZV 71654029 IC50 = 76700 nM T60857 C23PEW 71654030 IC50 = 16800 nM T60857 C5L7DG 71654095 IC50 > 30000 nM T60857 CCG4U7 71654098 IC50 = 5220 nM T60857 CG3M5N 71654183 IC50 = 43100 nM T60857 C0H7FK 71654184 IC50 = 13400 nM T60857 CR54BV 71654185 IC50 = 13600 nM T60857 C61MSA 71654187 IC50 = 33100 nM T60857 CI8OA5 71654189 IC50 = 38900 nM T60857 CIY17F 71654190 IC50 = 4900 nM T60857 CY1L0D 71654349 IC50 = 23300 nM T60857 C7CUQ8 71654350 IC50 = 5800 nM T60857 CFVE27 71716226 IC50 = 4960 nM T60857 CD35CT 71716837 IC50 = 15710 nM T60857 CV1D2T 71717010 IC50 = 8300 nM T60857 C6PEH3 71717460 IC50 = 5210 nM T60857 C4E0CJ 71717461 IC50 = 279 nM T60857 CQ02UI 71718049 IC50 = 120 nM T60857 CZ1UA2 71718050 IC50 = 290 nM T60857 C93TOG 71718051 IC50 = 22780 nM T60857 CHQ2S4 71718670 IC50 = 1080 nM T60857 CQ4I2G 71718851 IC50 = 51000 nM T60857 CR9Y7G 71719277 IC50 = 2230 nM T60857 CK52UZ 71719278 IC50 = 2400 nM T60857 CD7H8E 71720050 IC50 = 127800 nM T60857 CK9YE8 71720051 IC50 = 30200 nM T60857 CE7FC8 71720686 IC50 = 36900 nM T60857 CUGD52 71728326 IC50 = 770 nM T60857 C6BJ1A 71770556 IC50 = 790 nM T60857 CKDT91 71770679 IC50 = 13 nM T60857 CS3BP1 71770680 IC50 > 10000 nM T60857 CMXB37 73352188 IC50 = 2800 nM T60857 CHWS93 73671438 IC50 = 22 nM T60857 C4XV5A 73671439 IC50 = 12 nM T60857 CZ0R3F 73671440 IC50 = 10 nM T60857 CVU8K7 73671441 IC50 = 25 nM T60857 C4Q1FD 73671442 IC50 = 13 nM T60857 C17LVN 73671603 IC50 = 13 nM T60857 C7AW4O 73671604 IC50 = 460 nM T60857 CW2QZ6 76310104 IC50 > 30000 nM T60857 CD01GJ 76313800 IC50 = 3700 nM T60857 C7IC3Y 76313801 IC50 = 530 nM T60857 CDV56A 76317317 IC50 = 30000 nM T60857 C7MSO3 76317318 IC50 > 30000 nM T60857 CWE0U6 76317319 IC50 > 30000 nM T60857 C48FHA 76317320 IC50 = 4900 nM T60857 C3K0QB 76321039 IC50 > 30000 nM T60857 C3QU4Y 76321040 IC50 > 30000 nM T60857 CY1GW6 76321041 IC50 = 350 nM T60857 CVIJ82 76321042 IC50 = 2900 nM T60857 CTD09I 76321043 IC50 > 30000 nM T60857 CT9J3S 76321044 IC50 > 30000 nM T60857 C29DCS 76321045 IC50 > 30000 nM T60857 CA8B6L 76324692 IC50 = 9100 nM T60857 CB54FA 76324693 IC50 > 30000 nM T60857 CTSQ91 76328250 IC50 = 390 nM T60857 C10NVU 76328251 IC50 > 30000 nM T60857 C3WD7H 76328252 IC50 = 5520 nM T60857 C5B3DI 76328253 IC50 = 2300 nM T60857 C2NIF6 76328254 IC50 = 700 nM T60857 CE3TG2 76331929 IC50 > 30000 nM T60857 CI62UR 76331930 IC50 = 660 nM T60857 CH54NX 76331931 IC50 > 30000 nM T60857 C7GX8E 76334072 IC50 = 440 nM T60857 CYC73V 76335508 IC50 = 21900 nM T60857 CA34NL 76335509 IC50 > 30000 nM T60857 CI9R6D 76335510 IC50 > 30000 nM T60857 CBG41Z 90646227 IC50 = 8000 nM T60857 CD1LR5 101913702 IC50 = 110 nM T60857 C3UC1Z 101913703 IC50 = 110 nM T60857 CL28SZ 118714856 IC50 = 4500 nM T60857 CBLH92 118714857 IC50 = 970 nM T60857 CZC46M 118714858 IC50 = 2200 nM T60857 CEVP67 118714859 IC50 = 3100 nM T60857 CWLJ15 118714860 IC50 = 420 nM T60857 CF10SB 118714861 IC50 = 560 nM T60857 CZG5P4 118714862 IC50 = 1100 nM T60857 CUY16V 118714863 IC50 = 850 nM T60857 CHOR15 118714864 IC50 = 390 nM T60857 C8ZES0 118714865 IC50 = 320 nM T60857 C4HZ7W 118714866 IC50 = 220 nM T60857 CEZ9J4 118714867 IC50 = 360 nM T60857 C9IGN4 118714868 IC50 = 890 nM T60857 C10STI 118714869 IC50 = 570 nM T60857 CF83WX 118714870 IC50 = 160 nM T60857 CFJ76A 118714871 IC50 = 470 nM T60857 CHPF34 118714872 IC50 = 540 nM T60857 C58NMF 118714873 IC50 = 770 nM T60857 CMO7V6 118714874 IC50 = 910 nM T60857 CPB50U 118714875 IC50 = 400 nM T60857 CIR37V 118714876 IC50 = 540 nM T60857 C8KQ2S 118714877 IC50 = 580 nM T60857 CQC4I0 118714878 IC50 = 800 nM T60857 C39SRQ 118714879 IC50 = 840 nM T60857 CKZ2X3 118714880 IC50 = 960 nM T60857 C3XM9H 118800430 IC50 = 38000 nM T60857 CI4OQ5 122192740 IC50 = 57 nM T60857 CP90JH 122192741 IC50 = 86 nM T60857 CU96HS 122192742 IC50 = 35 nM T60857 C5Z4RW 122192743 IC50 = 36 nM T60857 CG6NF1 124464431 IC50 = 50 nM T60857 C5RFW4 129056873 IC50 = 1050 nM T60857 C8FDM7 129056875 IC50 = 820 nM T60857 C1MEO8 129056877 IC50 = 6000 nM T60857 CVM7K8 132473032 IC50 = 260 nM T60857 CCW36V 134131641 IC50 = 389.05 nM T60857 CAMG14 134139299 IC50 = 77.62 nM T60857 CGN6P0 134143813 IC50 = 41.69 nM T60857 CKA01N 134145805 IC50 = 1310 nM T60857 C1KAO0 134146656 IC50 = 25.12 nM T60857 C1SDT4 134149262 IC50 = 13 nM T60857 CW75QL 134157479 IC50 = 450 nM T60857 C2S0YD 134817174 IC50 = 63.1 nM T60857 C4D2AR 135304433 IC50 = 290 nM T60857 C9XI8T 135304436 IC50 = 130 nM T60857 C4IUR9 135304437 IC50 = 89 nM T60857 CSA5F0 135304444 IC50 = 110 nM T60857 CM9OG2 135304447 IC50 = 348 nM T60857 CPH27K 135304451 IC50 = 135 nM T60857 CB2Z1T 135304462 IC50 = 160 nM T60857 CBWN04 135304464 IC50 = 60 nM T60857 C1QB9U 135304477 IC50 = 300 nM T60857 CG5BK9 135304478 IC50 = 1800 nM T60857 CFK20G 135304481 IC50 = 110 nM T60857 C7JT0H 135304483 IC50 = 453 nM T60857 C8HO9M 135304484 IC50 = 156 nM T60857 C4YW6R 135304486 IC50 = 233 nM T60857 CT35VP 135304491 IC50 = 3600 nM T60857 C3R5EZ 135304495 IC50 = 94 nM T60857 CSMQ56 135304497 IC50 = 70 nM T60857 CK3IG5 135304499 IC50 = 2800 nM T60857 CBI16U 135304501 IC50 = 76 nM T60857 CJ45KT 135304509 IC50 = 140 nM T60857 C5AWQ4 135304510 IC50 = 1800 nM T60857 C1SV3F 135304513 IC50 = 100 nM T60857 CN2X9K 135304517 IC50 = 98 nM T60857 CHA53F 135304521 IC50 = 91 nM T60857 CO8E4J 135304524 IC50 = 135 nM T60857 C0BO7W 135304526 IC50 = 260 nM T60857 C21XJC 135304527 IC50 = 81 nM T60857 CI41GV 135304528 IC50 = 200 nM T60857 CI17MG 135304531 IC50 = 866 nM T60857 CH92PF 135304537 IC50 = 98 nM T60857 C2R5FK 135304538 IC50 = 110 nM T60857 CB5OL8 135304566 IC50 = 190 nM T60857 CN8P6S 135304567 IC50 = 125 nM T60857 CN2Y5T 135304571 IC50 = 200 nM T60857 CZ4HF6 135304587 IC50 = 370 nM T60857 CO31BZ 135304589 IC50 = 126 nM T60857 C52YBD 135304593 IC50 = 130 nM T60857 C6VI2Z 135304602 IC50 = 70 nM T60857 CS9CO6 135304832 IC50 = 330 nM T60857 CIDB04 135304925 IC50 = 180 nM T60857 CMBZ28 135304956 IC50 = 120 nM T60857 CRG5E6 135304958 IC50 = 88 nM T60857 C62OME 135304959 IC50 = 273 nM T60857 CQ73IA 135305074 IC50 = 132 nM T60857 C36PQU 135580289 IC50 = 1460 nM T60857 CY68HL 136236285 Ki = 118000 nM T60857 C10AZF 137349099 IC50 = 310 nM T60857 C4UE9D 137642579 IC50 = 470 nM T60857 CR10SV 137646927 IC50 = 1600 nM T60857 C2OQN1 138115373 IC50 = 300 nM T60857 C2OBN6 139188626 IC50 = 15000 nM T60857 C2EI4N 142412490 IC50 = 16000 nM T60857 C06AQB 142412524 IC50 = 6600 nM T60857 CDWX90 142412552 IC50 = 2300 nM T60857 CL3N0A 142412555 IC50 = 540 nM T60857 CZ26DS 142412606 IC50 = 1200 nM T60857 CLS26W 142412611 IC50 = 1000 nM T60857 C2AFV9 142412627 IC50 = 70 nM T60857 CK8T7Y 145951864 IC50 > 50000 nM T60857 CT89FP 145952913 IC50 >= 50000 nM T60857 C2DH1U 145953163 IC50 = 480 nM T60857 CN1W2C 145954680 IC50 > 50000 nM T60857 CMK21Q 145958984 IC50 = 32790 nM T60857 CTW1E5 145960123 IC50 = 1600 nM T60857 C91BHP 145971744 IC50 > 50000 nM T60857 CV2H4Q 145978951 IC50 = 213 nM T60857 C1EHA7 145979779 IC50 = 168 nM T60857 C5XJ0C 145980540 IC50 = 778 nM T60857 CWSU97 145981124 IC50 = 683 nM T60857 COI95A 145981258 IC50 = 480 nM T60857 C8K9ZI 145981397 IC50 = 730 nM T60857 CHM7A4 145983373 IC50 = 1410 nM T60857 CILB62 145984049 IC50 = 550 nM T60857 CN4O3U 145984086 IC50 = 190 nM T60857 CE1B9Z 145984193 IC50 = 400 nM T60857 CAQX10 145984948 IC50 = 3480 nM T60857 CJ34RC 145985588 IC50 = 310 nM T60857 CW38AP 145986388 IC50 = 1830 nM T60857 C8L9NI 145987501 IC50 = 7800 nM T60857 CM6PJ2 145988332 IC50 = 5540 nM T60857 CJ97BK 145988505 IC50 = 237 nM T60857 CW9RP2 145988662 IC50 = 160 nM T60857 CGZH45 145989229 IC50 = 684 nM T60857 CH4K8Y 145989901 IC50 = 5050 nM T60857 C3KBH8 145991531 IC50 = 676 nM T60857 C6MPJ4 145991600 IC50 = 278 nM T60857 C0MUT1 145992201 IC50 = 15500 nM T60857 CX3US2 145992914 IC50 = 287 nM T60857 CFS75D 145993116 IC50 = 255 nM T60857 C0L4TR 145993678 IC50 = 469 nM T60857 CH8J3B 145993940 IC50 = 510 nM T60857 CU81TG 155511105 IC50 = 23110 nM T60857 CYLC32 155513784 IC50 = 11690 nM T60857 CE0S8M 155516999 IC50 > 50000 nM T60857 CQK25N 155568033 IC50 = 940 nM T60857 D00DDO 268734 Ki = 4200 nM T60857 D00XMO 44126813 Ki = 20500 nM T60857 D03APP 4386 IC50 = 1500 nM T60857 D03POE 4044373 IC50 = 11000 nM T60857 D06SPO 9445 Ki = 94000 nM T60857 D06YGF 5281787 IC50 = 1700 nM T60857 D0DF1Z 19539 IC50 = 680 nM T60857 D0K9YS 44576211 IC50 = 13 nM T60857 D0MC5H 11009103 Ki = 33400 nM T60857 D0Q9RA 44126812 Ki = 16200 nM T60857 D0U4VL 5472440 Ki = 680 nM T60857 D0Z0IR 20313173 Ki = 69600 nM T63846 D04AHQ 71721540 IC50 = 390 nM T63846 D0E3TC 44259 IC50 = 59.3 nM T63846 D03BNU 59604787 IC50 > 10000 nM T63846 D0T3ME 156422 IC50 > 30000 nM T63846 CRC65X 9863786 IC50 > 30000 nM T63846 C8K9HL 10142476 Ki = 72 nM T63846 C8BHJ3 10226185 Ki = 374 nM T63846 C78SMB 10227510 Ki = 18 nM T63846 CXN06I 10227557 Ki = 608 nM T63846 C0SR5Y 10278151 Ki = 48 nM T63846 CACS26 11561968 Ki > 4000 nM T63846 CU0E8O 11690457 Ki = 2200 nM T63846 CM4F0B 21899142 Ki = 12 nM T63846 C7YG1N 24759534 IC50 < 10 nM T63846 CY8L7E 24896769 IC50 > 10000 nM T63846 CA75YC 25169380 IC50 = 293000 nM T63846 CC3BU0 25169381 IC50 = 96000 nM T63846 CFB65H 25169382 IC50 = 195000 nM T63846 CRXS80 25169384 IC50 = 175000 nM T63846 CRB74Z 44412281 IC50 = 750 nM T63846 C3VRO9 44557921 IC50 > 10000 nM T63846 CLS29B 46872626 IC50 > 10000 nM T63846 CD2K4R 50908681 Ki > 1000000 nM T63846 C8NA4L 53384644 IC50 > 30000 nM T63846 CO75VX 58056108 Ki = 400 nM T63846 C8CG6L 58056265 Ki = 2800 nM T63846 C8GFI0 58056341 Ki = 510 nM T63846 CXJ63M 59603829 IC50 = 19 nM T63846 CQEU96 59603842 IC50 = 9 nM T63846 COH62U 60097413 IC50 > 10000 nM T63846 C1MR8Q 60097495 IC50 > 10000 nM T63846 CV63UL 67240318 IC50 > 10000 nM T63846 CYI75G 68678653 IC50 > 30000 nM T63846 C5DGR9 69036886 IC50 = 10000 nM T63846 CYJ4C6 76955703 IC50 < 100 nM T63846 CSH9R0 77847460 IC50 < 100 nM T63846 CQ2SU8 78673832 IC50 > 30000 nM T63846 CE0W9R 78673833 IC50 > 30000 nM T63846 C1HW4B 89735655 IC50 = 1900 nM T63846 CX58DI 118716791 IC50 > 30000 nM T63846 CD9X2B 118716796 IC50 > 30000 nM T63846 C2YJ0O 118716797 IC50 > 30000 nM T63846 CL3UO9 118716798 IC50 > 30000 nM T63846 C71BAM 118716799 IC50 > 30000 nM T63846 CU4EL6 118716806 IC50 > 30000 nM T63846 CUS38N 127034643 IC50 = 900 nM T63846 CZD87E 127037084 IC50 = 14 nM T63846 CB9Z0V 127038973 IC50 = 15 nM T63846 C4Z5MQ 131839619 IC50 = 23 nM T63846 C7PJ6X 135566704 IC50 > 30000 nM T63846 CU0SZ4 136074298 IC50 < 100 nM T63846 CDMS84 136074299 IC50 < 100 nM T63846 CH3M4B 137083628 IC50 > 30000 nM T63846 CJA07O 137083629 IC50 > 30000 nM T63846 C9F8PX 137083630 IC50 > 30000 nM T63846 CS61AX 137659496 IC50 > 100000 nM T63846 CJ0G3C 138376590 Ki > 6100 nM T63846 C5J2WV 138728749 IC50 = 72 nM T63846 CVU63L 139582016 IC50 = 44 nM T63846 C8PH9S 139582017 IC50 = 27 nM T63846 C6VB3O 145925651 IC50 >= 5000 nM T63846 CX05ZN 145979845 IC50 = 21 nM T63846 CHX57D 155511560 Ki > 10000 nM T63846 C2MD1Q 155513187 IC50 > 10000 nM T63846 C17BHJ 155516763 IC50 > 10000 nM T63846 C08VAM 155517957 IC50 > 10000 nM T63846 C8UI7G 155520013 IC50 > 10000 nM T63846 CCL0S9 155520435 IC50 > 10000 nM T63846 CWP05R 155527255 Ki > 5500 nM T63846 CE2YX6 155527737 Ki = 4700 nM T63846 CSJB85 155530835 Ki = 95 nM T63846 CL5F3C 155537218 Ki = 24 nM T63846 CG4LQ2 155539650 Ki = 340 nM T63846 CX9FM8 155548286 IC50 > 10000 nM T63846 CM8O9G 155552851 Ki = 5400 nM T63846 CWO25P 155555362 Ki = 500 nM T63846 C4Y6BV 155556454 Ki > 5700 nM T63846 CWJ08R 155560232 Ki = 190 nM T63846 C3D2GP 155562155 IC50 = 6943 nM T63846 D00ERW 44444843 Ki = 3011 nM T63846 D04ZIV 58056241 IC50 = 55 nM T63846 D0I2FZ 11983295 IC50 = 300 nM T63846 D0J3LR 11634725 Ki > 10000 nM T63846 D0J8VR 25169383 IC50 = 23000 nM T63846 D0T2NE 58056092 IC50 = 983 nM T89034 D05EAM 4735 IC50 = 3600 nM T89034 D05HXX 5526 IC50 = 3100 nM T89034 D05PHH 3447 IC50 = 1550 nM T89034 D07UWV 92722 Ki = 257000 nM T89034 D07XHO 4413 IC50 = 240 nM T89034 D08YIN 1727 Ki > 2000000 nM T89034 D0FD0H 564 IC50 = 105000 nM T89034 D0I0RJ 16231 IC50 > 20000 nM T89034 D0J0BU 10275777 IC50 > 10000 nM T89034 D0M7JT 216210 Ki = 1695 nM T89034 D0V3YT 10324367 IC50 > 100000 nM T89034 D0X9CH 3010818 IC50 = 8700 nM T89034 D00LOB 9866964 Ki > 26000 nM T89034 D01MUU 183797 Ki = 700 nM T89034 D02ALZ 127139 Ki = 310 nM T89034 D0I7MX 9871765 Ki = 7400 nM T89034 D0ID3W 9911502 IC50 > 158000 nM T89034 D0PK7J 56599309 Ki = 0.77 nM T89034 D02INZ 2387 Ki = 2650 nM T89034 D02QTV 122267 IC50 = 670 nM T89034 D08INO 9895194 Ki = 1200 nM T89034 D0D5RH 11641515 IC50 > 60000 nM T89034 D0GR2H 11740077 IC50 = 41000 nM T89034 D0S2JG 9913629 Ki = 47900 nM T89034 D0Y5EX 122296 Ki = 5.1 nM T89034 C71WRJ 1503 Ki = 25000 nM T89034 CY5B9C 1504 Ki = 5000 nM T89034 C2KE5Q 1508 Ki = 12000 nM T89034 CKO7V4 1701 IC50 = 240000 nM T89034 C7BU1L 2138 Ki = 12589.25 nM T89034 C4S1PB 4300 Ki > 75000 nM T89034 CL1T7V 4301 Ki = 90000 nM T89034 C3GXF8 5713 IC50 = 530 nM T89034 C0YU1V 16157 Ki = 2610000 nM T89034 CT28FD 80002 Ki < 10000000 nM T89034 COHM79 117475 Ki = 3981071.71 nM T89034 CMG15V 122129 Ki = 11000 nM T89034 CK9AZ0 122670 Ki = 112000 nM T89034 C50XVJ 159772 Ki < 10000000 nM T89034 C1BHS3 193409 Ki = 51000 nM T89034 CD14RN 197789 Ki = 100000 nM T89034 CZP0Y1 204101 Ki > 15000 nM T89034 CU4G3Y 309369 Ki = 19952.62 nM T89034 CIR92Q 409363 Ki < 10000000 nM T89034 C32CWP 409364 Ki < 10000000 nM T89034 CZ17HE 445157 Ki = 30000 nM T89034 C2Z0XW 445482 Ki = 2300 nM T89034 CU6X2A 445847 Ki = 2700 nM T89034 C5UX1L 447478 Ki = 310 nM T89034 CVND42 447482 Ki = 1300 nM T89034 C4OKV5 447486 Ki = 2200 nM T89034 CC9G5O 447490 Ki = 1100 nM T89034 CR2DX3 447496 Ki = 1700 nM T89034 COYS31 447502 Ki = 21000 nM T89034 CVI28M 447508 Ki = 600 nM T89034 CS09BE 447510 Ki = 3200 nM T89034 C87GLP 447540 Ki = 2600 nM T89034 C87OTC 447733 Ki = 16000 nM T89034 CF6D4B 447734 Ki = 498 nM T89034 CHT05K 447735 Ki = 768 nM T89034 C5FG9U 448513 Ki = 630957.34 nM T89034 CFMI91 448548 Ki = 11000 nM T89034 C5QKC3 448605 Ki = 150 nM T89034 CX5MS1 448610 Ki = 3800 nM T89034 CO01KD 456168 Ki = 8190 nM T89034 C0P9RD 459983 Ki = 8180 nM T89034 C3NB2K 459984 Ki = 3830 nM T89034 C2J3VS 576480 Ki = 316227.77 nM T89034 C49RWG 1549311 Ki < 10000000 nM T89034 CNBW97 2250229 IC50 < 1000 nM T89034 C4ZUJ5 2757788 Ki < 50000 nM T89034 CTE79D 3011892 Ki > 50000 nM T89034 C40DHV 3016780 Ki = 1584893.19 nM T89034 CU43OY 3088969 Ki > 50000 nM T89034 CB58JC 3357702 Ki = 251188.64 nM T89034 CZ9ST3 3564407 Ki = 316227.77 nM T89034 C1DU3P 3580940 Ki < 10000000 nM T89034 CIR7L6 3621644 Ki < 10000000 nM T89034 C5PJK7 3631189 Ki < 10000000 nM T89034 CQY92E 3660962 IC50 = 240000 nM T89034 C7ZTI9 3676069 Ki = 398107.17 nM T89034 CCS5F4 4475490 Ki = 10200 nM T89034 C13DFJ 4475491 Ki = 8400 nM T89034 C8EK6S 4620241 Ki = 7943282.35 nM T89034 CV89RH 4713317 Ki = 12000 nM T89034 C2UD9T 4713319 Ki = 5000 nM T89034 CV8W5G 4713320 Ki = 7800 nM T89034 C60OCJ 4713322 Ki = 55000 nM T89034 CRK73Q 4713323 Ki = 12000 nM T89034 CQC05H 4713327 Ki = 6400 nM T89034 CJC7N6 4713329 Ki = 2600 nM T89034 CY5KR6 4713353 Ki = 7700 nM T89034 C9A0IZ 4713356 Ki = 7000 nM T89034 CVT61D 4713357 Ki = 4000 nM T89034 CD02VO 4713366 Ki = 1400 nM T89034 C2G7OB 4713372 Ki = 400 nM T89034 C81KBP 4713415 Ki = 8200 nM T89034 CMR9D1 4713416 Ki > 1000000 nM T89034 CV95FQ 5108695 Ki = 316227.77 nM T89034 CHF96N 5173985 Ki < 10000000 nM T89034 CG7BH6 5221300 Ki = 3162277.66 nM T89034 CH0JF4 5280417 IC50 = 1500 nM T89034 C8I0VG 5289529 Ki = 8500 nM T89034 CQ26VM 5289531 Ki = 440 nM T89034 CLU8P2 5318214 IC50 = 2300 nM T89034 C1DR3H 6475892 IC50 = 13000 nM T89034 CN2B6S 6852211 Ki = 600 nM T89034 CX34ZD 9549214 Ki > 1800 nM T89034 C6JDM9 9799627 Ki = 1120 nM T89034 C2FHU7 9801905 IC50 = 1500 nM T89034 CKA6C4 9802514 Ki = 39000 nM T89034 C1FIN6 9804775 IC50 > 130 nM T89034 C6JIT7 9806444 IC50 > 11000 nM T89034 CAG59M 9808035 Ki = 4700 nM T89034 CH9IE6 9808346 Ki > 100000 nM T89034 C2AXV0 9809479 Ki > 15000 nM T89034 C8UX0O 9810198 Ki > 1000000 nM T89034 CF9S0B 9815838 Ki = 176500 nM T89034 CKN89B 9822176 Ki = 6900 nM T89034 C1D4EC 9822928 Ki = 14000 nM T89034 CPB20R 9826345 Ki = 1800 nM T89034 CS1DL7 9826716 IC50 = 43000 nM T89034 CB82VS 9827306 IC50 > 11000 nM T89034 CGN48U 9827867 IC50 > 2500 nM T89034 CP2X5B 9829453 Ki = 25000 nM T89034 C8Z5TX 9843775 Ki > 100000 nM T89034 C53JFK 9844392 Ki = 78200 nM T89034 C6VAG8 9845526 IC50 = 66000 nM T89034 C5Z2RH 9848091 IC50 > 11000 nM T89034 CL6QS0 9868922 Ki = 540 nM T89034 CIL85V 9871029 IC50 > 11000 nM T89034 C6ZB3K 9872552 IC50 > 11000 nM T89034 C87SWZ 9872983 Ki > 1000000 nM T89034 C5LV1Z 9873979 IC50 = 143000 nM T89034 CA9Z4S 9875345 Ki = 494000 nM T89034 CQP0V2 9886960 Ki = 290 nM T89034 C17NPU 9890541 IC50 > 2500 nM T89034 C1M2PU 9892103 IC50 > 11000 nM T89034 CNJ0W1 9893177 IC50 = 3270 nM T89034 C9SJ3T 9894908 IC50 = 1040 nM T89034 CKDP84 9895193 Ki = 390 nM T89034 C6PSQ7 9896889 Ki = 700000 nM T89034 CD5LQ0 9910982 Ki > 200000 nM T89034 C13XPD 9912856 Ki = 40000 nM T89034 C1C3VT 9914538 IC50 > 11000 nM T89034 CC0D5H 9915041 Ki > 15000 nM T89034 CFO1K9 9922130 Ki > 1000000 nM T89034 CLZ53G 9922131 Ki > 1000000 nM T89034 C2UX6D 9930716 Ki = 16000 nM T89034 C9I2ES 9931785 IC50 = 5800 nM T89034 CB7VR2 9934590 IC50 = 150 nM T89034 CG3B1P 9935390 Ki = 1700 nM T89034 CNE25D 9935474 Ki = 65000 nM T89034 C1XT2Y 9935746 Ki > 60000 nM T89034 CL2NV0 9935925 IC50 = 330 nM T89034 C5KS0R 9936020 IC50 > 11000 nM T89034 C49DRC 9936691 IC50 > 11000 nM T89034 C8F5CW 9937921 Ki > 35000 nM T89034 C8LR4T 9938917 Ki > 15000 nM T89034 CDT95S 9939426 Ki = 1460 nM T89034 CFK05S 9949275 Ki = 14500 nM T89034 C1RHT8 9949886 Ki = 250 nM T89034 CYP6S7 9952109 Ki = 27000 nM T89034 CW7TZ6 9953704 IC50 = 1460 nM T89034 C0R4GE 9954812 IC50 = 13000 nM T89034 CX85LD 9954980 Ki > 22000 nM T89034 C3EPC4 9955758 Ki > 22000 nM T89034 CCQE85 9956843 Ki > 30000 nM T89034 CYLI95 9956922 Ki = 32000 nM T89034 CBC2K3 9959749 IC50 > 11000 nM T89034 C0TV8Q 9962561 Ki = 212000 nM T89034 C5SA7F 9983043 IC50 > 2500 nM T89034 C1XJ9Y 9986673 IC50 = 800 nM T89034 CKIP10 9987251 IC50 = 2000 nM T89034 C8I7YZ 10006319 IC50 = 94 nM T89034 C7LWC0 10009777 IC50 = 68 ug.mL-1 T89034 CBL8D4 10026170 Ki = 170 nM T89034 CF1V4K 10027758 Ki > 7300 nM T89034 CX4TI5 10029172 Ki = 10900 nM T89034 C3E4DR 10029213 IC50 = 91000 nM T89034 C08PUS 10051441 IC50 = 81 nM T89034 CFCT67 10053115 Ki = 1200 nM T89034 C9KC6Q 10053945 IC50 = 10000 nM T89034 CXZ2V3 10054210 Ki = 300 nM T89034 C8YHP3 10055497 Ki = 287000 nM T89034 CBV7N2 10070407 IC50 = 370 nM T89034 CF4R2W 10074230 IC50 = 98 nM T89034 C9ZCS2 10074922 IC50 = 85 nM T89034 C7CW1P 10080504 IC50 > 10000 nM T89034 CR0ZL7 10091675 IC50 = 39000 nM T89034 CZH3W7 10094378 Ki > 200000 nM T89034 CQP65H 10095093 Ki = 57000 nM T89034 C3OG5U 10095865 IC50 > 20000 nM T89034 C17CDJ 10096845 IC50 = 367 nM T89034 CQB1V2 10101474 IC50 = 0.3 ug.mL-1 T89034 CW4RZ5 10116936 IC50 > 450 nM T89034 C1VT4F 10117027 Ki > 200000 nM T89034 C5E0SY 10126451 Ki = 1046 nM T89034 CR03NV 10131788 Ki > 1000000 nM T89034 CS2G4T 10140847 Ki = 56 nM T89034 C31QAL 10143532 Ki > 15000 nM T89034 C7L5IJ 10157296 Ki = 320 nM T89034 CL7U8P 10181581 Ki = 811 nM T89034 C7PC2K 10185292 IC50 > 170 nM T89034 CO51ZR 10205659 IC50 > 10000 nM T89034 CEP79T 10216518 Ki = 594 nM T89034 CC2EA1 10219529 Ki = 245000 nM T89034 C8V1AY 10225952 Ki = 53 nM T89034 C2XHG8 10248900 Ki = 10800 nM T89034 C4Z1LU 10255253 Ki > 7300 nM T89034 CS4F5P 10256448 IC50 = 68000 nM T89034 C4WV1A 10257345 IC50 = 869 nM T89034 C2F4TQ 10259285 Ki = 62200 nM T89034 CSX60M 10264543 Ki = 466000 nM T89034 CQ9ZO1 10275412 Ki > 28000 nM T89034 C0J1TD 10278414 Ki = 90 nM T89034 CNAX45 10287785 Ki = 955 nM T89034 CZM97W 10293977 Ki = 210000 nM T89034 C5EDW1 10294146 Ki = 400 nM T89034 C0T3CN 10296435 IC50 > 100000 nM T89034 CV10CU 10297977 IC50 > 10000 nM T89034 C1AP6H 10298858 IC50 > 10000 nM T89034 C4Q3TL 10322647 IC50 = 620000 nM T89034 C8SQ1N 10324263 Ki > 60000 nM T89034 C41ZLB 10326602 IC50 = 730 nM T89034 CP64HV 10342843 Ki = 744000 nM T89034 CK9J7X 10343728 IC50 > 25100 nM T89034 CF9Q3K 10345602 Ki > 200000 nM T89034 C10ISY 10367012 Ki = 165000 nM T89034 CJWE07 10368488 IC50 = 150 nM T89034 C67JPL 10370341 IC50 = 530 nM T89034 CNJ03F 10374840 Ki < 10000000 nM T89034 C26CSM 10386393 IC50 = 490 nM T89034 CSC52L 10390341 Ki = 5200 nM T89034 C8EPN7 10390481 Ki > 200000 nM T89034 CXF20B 10391310 IC50 = 36000 nM T89034 C6S4CO 10391715 Ki > 60000 nM T89034 C56NXW 10409551 IC50 = 660000 nM T89034 CB4X5P 10417378 Ki = 6 nM T89034 CJTH60 10432907 Ki = 966 nM T89034 C6AZ8B 10435038 Ki = 27000 nM T89034 CS80VR 10438758 Ki = 3000000 nM T89034 C4XD5V 10439687 Ki = 310000 nM T89034 C9HI6A 10460541 IC50 > 2500 nM T89034 CI87FD 10460564 IC50 = 726 nM T89034 C6KJM2 10461790 Ki > 50000 nM T89034 CU97PJ 10464707 IC50 = 12200 nM T89034 CWG91R 10472893 Ki = 32100 nM T89034 C63GRO 10479438 IC50 = 1240 nM T89034 CCP2N8 10480374 Ki > 7300 nM T89034 CV0X6G 10480463 IC50 > 11000 nM T89034 CG18KR 10483116 Ki > 86000 nM T89034 CEI65Z 10483775 Ki = 910 nM T89034 CFP53Y 10502109 IC50 > 33000 nM T89034 CS9NE0 10505479 IC50 = 45000 nM T89034 CT41HV 10509499 IC50 < 50000 nM T89034 C5ED3G 10529121 Ki = 113000 nM T89034 CLR6E5 10531398 Ki = 11000 nM T89034 CHP5F9 10554949 Ki = 2600 nM T89034 CU8N3V 10578280 Ki = 4900 nM T89034 C9UWZ7 10579207 Ki = 2300 nM T89034 C5W1VA 10579727 Ki = 3000 nM T89034 C2T4KP 10598728 IC50 = 7500 nM T89034 CCG70Y 10603018 Ki = 14000 nM T89034 C02RUZ 10603715 Ki = 19000 nM T89034 CC8DQ0 10604342 Ki = 11000 nM T89034 C8SUZ9 10624948 Ki = 52000 nM T89034 CEJ14F 10624997 Ki = 3300 nM T89034 CM1B3D 10626862 Ki = 7200 nM T89034 CV31AX 10628055 Ki = 100000 nM T89034 CFNH06 10645807 IC50 = 21000 nM T89034 CR5EX8 10648196 Ki = 19000 nM T89034 CPWH69 10648370 Ki = 30000 nM T89034 CKNW85 10648867 Ki = 29000 nM T89034 CD2X1K 10652683 IC50 < 50000 nM T89034 CBT96N 10664145 Ki = 400000 nM T89034 CJG9H6 10669349 Ki = 691000 nM T89034 CW1G9B 10672666 IC50 > 10000 nM T89034 C5VB1U 10695159 Ki > 1000000 nM T89034 CP4QC5 10696511 Ki = 414000 nM T89034 CGYR23 10696955 Ki = 5200 nM T89034 CGP79W 10697355 IC50 = 240 nM T89034 CK84UR 10697371 Ki = 2800 nM T89034 CK2C1R 10698387 Ki = 10200 nM T89034 CY2K8L 10699089 Ki = 15000 nM T89034 CSK62G 10717029 IC50 = 710 nM T89034 CPGV87 10718240 Ki > 1000000 nM T89034 CIKF89 10719580 Ki = 176000 nM T89034 CI7GB2 10721554 Ki = 3500 nM T89034 CU6T3H 10723324 Ki = 5000 nM T89034 CL7RC5 10742017 IC50 = 33000 nM T89034 CZ0Q8K 10742217 Ki = 152000 nM T89034 C7RWD8 10744643 Ki = 244000 nM T89034 C0RYX4 10744937 Ki = 2500 nM T89034 CKOQ35 10767421 Ki = 160000 nM T89034 CKU82G 10791027 IC50 = 6100 nM T89034 CXLS49 10791461 IC50 = 4300 nM T89034 CQB03L 10793925 Ki = 30000 nM T89034 CWVK42 10814863 IC50 = 3900 nM T89034 C3IN8W 10815545 Ki = 21000 nM T89034 CVQE76 10816339 Ki = 9000 nM T89034 CA25LK 10816909 Ki = 7800 nM T89034 CMCW41 10840061 Ki = 8600 nM T89034 CB86VA 10840391 Ki = 14000 nM T89034 CW7Q2U 10895700 IC50 > 250000 nM T89034 CQTC02 10903566 Ki = 5500 nM T89034 C8OA1L 10946869 Ki = 26000 nM T89034 C43SNO 11004109 Ki = 900 nM T89034 CC39SB 11009950 Ki = 350000 nM T89034 CYZL25 11015002 Ki = 350 nM T89034 CD9WJ8 11057540 Ki = 290 nM T89034 C2Y6VW 11057779 Ki = 190 nM T89034 C3HNB2 11068806 Ki = 2100 nM T89034 CT5I6N 11118898 IC50 = 146000 nM T89034 CAD15G 11149953 Ki = 5560 nM T89034 CJ4X7R 11158066 IC50 = 10800 nM T89034 C6LVG4 11186243 Ki = 3820 nM T89034 CTX9F3 11188793 Ki = 1190 nM T89034 CGC9O1 11227852 IC50 = 32200 nM T89034 CLA93S 11237163 Ki > 22000 nM T89034 CHLK70 11244460 Ki = 1970 nM T89034 CRDU42 11271947 Ki > 33000 nM T89034 CX9Z7A 11277660 IC50 > 250000 nM T89034 C86DZB 11292119 Ki = 631 nM T89034 C91GMZ 11317532 Ki > 100000 nM T89034 C6CDN3 11347670 Ki = 3870 nM T89034 CLY5G8 11350400 Ki = 765 nM T89034 CR8NW9 11351302 Ki > 22000 nM T89034 CTJ1Z2 11361949 Ki = 833 nM T89034 CGW75B 11419694 Ki = 33000 nM T89034 CIQH43 11445130 IC50 = 4900 nM T89034 C9O4NF 11450922 IC50 = 13000 nM T89034 C63LIR 11473486 Ki = 554 nM T89034 CJZ09N 11512593 Ki = 3700 nM T89034 C28BMR 11513105 Ki = 4100 nM T89034 CRNU10 11534959 Ki = 330 nM T89034 CD1A6T 11542037 Ki = 880 nM T89034 CA8KD7 11542038 Ki = 440 nM T89034 CBP69L 11557024 Ki = 5000 nM T89034 CCG84F 11563457 Ki = 780 nM T89034 CV46NL 11563632 Ki = 10200 nM T89034 CEAZ46 11569930 Ki = 730 nM T89034 C3TJ7M 11570580 Ki = 2000 nM T89034 C6RHD8 11570700 Ki = 2800 nM T89034 C1DN2L 11570759 Ki = 4200 nM T89034 C6FG8V 11577055 Ki = 1400 nM T89034 CIY34V 11577968 Ki = 2500 nM T89034 CJ38EP 11577970 Ki = 3400 nM T89034 C7MF9N 11578158 Ki = 1000 nM T89034 CTSK74 11584729 Ki = 2400 nM T89034 C1RQ6P 11592130 Ki = 2500 nM T89034 CBC84M 11592593 Ki = 640 nM T89034 C7ZS8L 11592600 Ki = 3200 nM T89034 C7QTY8 11606981 Ki = 1800 nM T89034 CU07NO 11607091 Ki = 1300 nM T89034 CL9TZ2 11614477 Ki = 1800 nM T89034 CB4O2Q 11621579 Ki = 1400 nM T89034 CD3R1E 11627899 Ki = 4500 nM T89034 CB9P0Q 11628768 Ki = 1200 nM T89034 CO3Q9N 11635973 Ki = 820 nM T89034 CRX98P 11636026 Ki = 7200 nM T89034 CW10CL 11642802 Ki = 1400 nM T89034 C2W5XF 11656797 Ki = 1200 nM T89034 C4SAR0 11657278 Ki = 6000 nM T89034 CVQ16C 11664107 Ki = 1200 nM T89034 CPZG49 11664334 Ki = 12000 nM T89034 CT9E0G 11664643 Ki = 1400 nM T89034 CWV87X 11671266 Ki = 2700 nM T89034 CE0A6N 11671776 Ki = 360 nM T89034 C85GCY 11671956 Ki = 260 nM T89034 C1DHO6 11678360 Ki = 210 nM T89034 C4IBO3 11678764 Ki = 1400 nM T89034 CJP9O1 11684611 Ki = 8400 nM T89034 C69YSR 11693028 Ki = 940 nM T89034 CCQY30 11693049 Ki = 3100 nM T89034 CPFW75 11699600 Ki = 1700 nM T89034 C3VS2H 11699903 Ki = 840 nM T89034 CNV09Z 11699913 Ki = 760 nM T89034 CKQ4O2 11721188 Ki = 2800 nM T89034 C4UB2X 11721375 Ki = 3100 nM T89034 CQ5U8H 11739438 Ki = 1030 nM T89034 CNPT36 11756005 Ki = 210000 nM T89034 C7JLR1 11774107 Ki = 1060 nM T89034 CR2E9T 11782463 Ki = 250 nM T89034 CQK1D6 11796882 IC50 = 90 ug.mL-1 T89034 CNO67W 11798089 Ki = 57000 nM T89034 C7WYH2 11801086 Ki = 18000 nM T89034 C2G7KQ 11802399 Ki = 420000 nM T89034 CPJS89 11811066 Ki > 500000 nM T89034 C98ZOR 11824040 Ki = 26000 nM T89034 CPR4I1 12047383 Ki = 4000 nM T89034 C5U0FJ 12047384 Ki = 6200 nM T89034 C5FU3H 12047385 Ki = 109000 nM T89034 CV23RM 12181440 Ki = 16900 nM T89034 CZ15UV 12253678 Ki < 10000000 nM T89034 CJL46R 12254250 Ki = 125892.54 nM T89034 C3OHB0 12336481 Ki < 10000000 nM T89034 CX9Q2G 12420538 Ki < 10000000 nM T89034 C5PVL9 12456162 Ki = 1000000 nM T89034 CBDW65 12459438 Ki = 3900 nM T89034 CYRN35 14082458 IC50 = 700000 nM T89034 C20YIT 14082554 IC50 = 69000 nM T89034 CLD34I 14082564 IC50 = 30000 nM T89034 C94BTA 14346967 Ki < 10000000 nM T89034 C54OBM 15101654 IC50 = 12000 nM T89034 CS0QX7 15101655 IC50 = 15000 nM T89034 C1H2GY 15101698 IC50 = 200000 nM T89034 CP35QH 15227625 Ki > 500000 nM T89034 CBVA60 15227963 Ki > 500000 nM T89034 CB91UM 15227967 Ki > 500000 nM T89034 CP63GF 15534822 IC50 > 2500 nM T89034 C7VH6K 15950345 Ki > 27000 nM T89034 C2QO1B 15955412 Ki > 50000 nM T89034 C19ARJ 15984063 Ki = 430 nM T89034 CA8Y1K 16046152 Ki > 15000 nM T89034 CNBJ60 16046153 Ki > 15000 nM T89034 C5TBL6 16049247 IC50 = 13000 nM T89034 C9BH4X 16086308 IC50 = 1900 nM T89034 CF1V2N 16086310 IC50 = 15000 nM T89034 C9JX7U 16086312 IC50 = 1540 nM T89034 CK7IM0 16086316 IC50 = 900 nM T89034 CT9QM5 16086318 IC50 = 8000 nM T89034 CXO65R 16086320 IC50 = 4200 nM T89034 C3EUJ6 16086336 IC50 = 37 nM T89034 CR9EN3 16086338 IC50 = 990 nM T89034 CR7B3D 16086340 IC50 = 10000 nM T89034 C90CXM 16086342 IC50 = 1700 nM T89034 C7T5AI 16086344 IC50 = 900 nM T89034 CJZ63N 16086346 IC50 = 5000 nM T89034 C05XAN 16086348 IC50 = 7200 nM T89034 CACN42 16086349 IC50 = 900 nM T89034 CO8GZ6 16156362 Ki = 2700 nM T89034 CA0Y5E 16219042 Ki = 501187.23 nM T89034 CN6CJ2 16220264 IC50 = 340 nM T89034 CZB89F 16657876 Ki = 16000 nM T89034 CS9W6K 16657879 Ki = 45000 nM T89034 C09DTL 16657882 Ki > 100000 nM T89034 CBPA54 16658031 Ki = 41000 nM T89034 C7JHS4 16658108 Ki = 71000 nM T89034 C6V7DS 16658181 Ki > 100000 nM T89034 C0TW3X 16658183 Ki > 100000 nM T89034 CPNJ21 16658250 Ki > 100000 nM T89034 C5Q6JS 16658289 Ki > 100000 nM T89034 CG98OH 16658290 Ki > 100000 nM T89034 CO3ZV4 16658354 Ki > 30000 nM T89034 C46CDF 16658356 Ki = 9800 nM T89034 C8DI4G 16658357 Ki > 100000 nM T89034 C0Y4ZW 16658407 Ki > 100000 nM T89034 C6NR2O 16658408 Ki = 23000 nM T89034 CB6PC9 16658409 Ki = 15000 nM T89034 CBX83S 16658633 Ki > 100000 nM T89034 CZ58FK 16658680 Ki > 30000 nM T89034 C70XKG 16658742 Ki > 100000 nM T89034 CQDT69 16658745 Ki > 100000 nM T89034 CU60AH 16718671 IC50 = 57000 nM T89034 COAB94 16718712 IC50 = 16000 nM T89034 CU28CE 16718713 IC50 = 2800 nM T89034 CLI4D7 16718757 IC50 = 2000 nM T89034 C2SFC0 16718759 IC50 = 1200 nM T89034 CC20PS 16718760 IC50 = 11000 nM T89034 CCKO80 16718762 IC50 = 1200 nM T89034 CTZ74D 16718807 IC50 = 14000 nM T89034 C37MRI 16718808 IC50 = 3000 nM T89034 C87WGF 17750368 Ki > 500000 nM T89034 CB6R1Z 17809213 IC50 = 14.37 nM T89034 CTQ85L 18397340 Ki > 1000000 nM T89034 CZ4L5C 18397341 Ki > 1000000 nM T89034 CU5N8E 18397342 Ki = 632000 nM T89034 C4HE7G 18397344 Ki = 60000 nM T89034 CF1Y7P 18397345 Ki > 1000000 nM T89034 C3D1VS 18397346 Ki = 66000 nM T89034 CEJ3K1 18397347 Ki > 1000000 nM T89034 CVB47A 18397350 Ki > 1000000 nM T89034 C7DB0W 18397352 Ki = 134000 nM T89034 C03OYT 18397353 Ki > 1000000 nM T89034 CP3ZL0 18397354 Ki > 1000000 nM T89034 CM28UY 18397357 Ki > 1000000 nM T89034 C0POA1 18397359 Ki > 1000000 nM T89034 CSW0L3 18397360 Ki > 1000000 nM T89034 CN9S6X 18397370 Ki > 1000000 nM T89034 CS21RN 18397380 Ki > 1000000 nM T89034 CYO70H 18545754 Ki > 1000000 nM T89034 C9NB0Z 18675062 IC50 = 38000 nM T89034 C29WYS 18675086 IC50 = 8400 nM T89034 CK6U1I 18675238 IC50 = 2200 nM T89034 CN0LW2 18675252 IC50 = 25000 nM T89034 CD9UE4 18675298 IC50 = 12000 nM T89034 CF4W5D 18727604 IC50 > 10000 nM T89034 CB0IQ4 18727607 IC50 > 11000 nM T89034 C31ZAL 18727831 IC50 > 11000 nM T89034 CJY67O 18727833 IC50 > 11000 nM T89034 C02HEA 18727834 IC50 > 11000 nM T89034 CJSL38 18727836 IC50 > 11000 nM T89034 C8AMY9 18727838 IC50 > 11000 nM T89034 CY8AC3 18727841 IC50 > 11000 nM T89034 CD02TK 18727852 IC50 > 11000 nM T89034 C1JMX5 18727855 IC50 > 11000 nM T89034 CX36SV 18771291 Ki = 4100 nM T89034 C24CAY 18771297 Ki = 68000 nM T89034 CAZ56G 19388089 Ki > 500000 nM T89034 CK71LJ 19841587 Ki < 10000000 nM T89034 CBD5Y9 20229530 Ki = 60000 nM T89034 CO2JG4 20595081 IC50 > 11000 nM T89034 CM7BH1 20595091 IC50 > 11000 nM T89034 CCH5N1 20595225 IC50 > 11000 nM T89034 CXH09O 20631502 IC50 = 0.229 nM T89034 C7LHE8 20641745 IC50 = 6960 nM T89034 CZ6KH9 20760195 Ki > 15000 nM T89034 C2Z9NT 21192495 Ki = 3000 nM T89034 CLT36V 21250176 IC50 = 53000 nM T89034 CGC48U 21250249 IC50 = 14800 nM T89034 CRYB96 21250293 IC50 = 60000 nM T89034 CLV49W 21250386 IC50 > 100000 nM T89034 CN2YE9 21250416 IC50 = 69000 nM T89034 CRD4V1 21250427 IC50 = 72000 nM T89034 C9H7ZI 21250518 IC50 = 75000 nM T89034 CNTI15 21366511 IC50 > 11000 nM T89034 C5S8ZW 21366513 IC50 > 11000 nM T89034 C67QCO 21366574 IC50 > 11000 nM T89034 CS2L1Y 21366575 IC50 > 11000 nM T89034 CX1WM9 21366579 IC50 > 11000 nM T89034 CA07SQ 21434854 Ki < 10000000 nM T89034 CA63IO 21706943 Ki = 6000 nM T89034 C80JYP 21707001 Ki = 9400 nM T89034 C3H6XW 21707065 Ki = 3523 nM T89034 C5JD2U 21707080 Ki = 6600 nM T89034 CI0SJ2 21967345 Ki > 7300 nM T89034 CF4JN6 22010099 Ki > 1000000 nM T89034 C7ZA4U 22010100 Ki > 1000000 nM T89034 CFO41P 22010118 Ki = 3000 nM T89034 CNOT37 22098976 Ki < 10000000 nM T89034 C1R9CX 22336133 IC50 = 0.127 nM T89034 CHOQ30 22336142 IC50 = 0.913 nM T89034 CVG29W 22336143 IC50 = 0.252 nM T89034 CB7N4X 22336146 IC50 = 1.066 nM T89034 C5O7VB 22336151 IC50 = 0.035 nM T89034 CTOR48 22336172 IC50 = 0.408 nM T89034 C51FCG 22336174 IC50 = 0.494 nM T89034 CXZ92L 22336180 IC50 = 2.47 nM T89034 CDZ64O 22498328 IC50 > 100000 nM T89034 C4YL7S 22556963 Ki = 1500 nM T89034 C9VXC8 22556983 Ki = 4600 nM T89034 CA3N9L 22883564 Ki = 5800 nM T89034 C1R0UD 22883585 Ki > 7300 nM T89034 C13-JAN 22883594 Ki = 1500 nM T89034 CQ70HF 23586156 IC50 = 201 nM T89034 CRX19I 23646295 Ki > 15000 nM T89034 CCRD27 23646312 Ki > 25000 nM T89034 C1WE6B 23646315 Ki > 15000 nM T89034 CSFH79 23646622 Ki = 4400 nM T89034 C35HJA 23646623 Ki = 5500 nM T89034 C7E4SA 23646732 Ki = 1000 nM T89034 C9ZJ4W 23655167 IC50 = 78000 nM T89034 CKH4O5 24180463 Ki > 22000 nM T89034 C7AYO1 24748789 IC50 = 125000 nM T89034 CVO5L6 24748791 IC50 = 6200 nM T89034 CUAY58 24749175 IC50 = 900 nM T89034 CL2PU5 24750417 IC50 = 17000 nM T89034 CJSO87 24849206 Ki > 33000 nM T89034 CZI85G 24984725 Ki = 1.1 nM T89034 CN0ZW3 24999867 Ki > 27000 nM T89034 CEM32W 25001205 Ki = 3400 nM T89034 CAO2V4 25030840 Ki = 1300 nM T89034 CU82IO 25030929 Ki = 500 nM T89034 C7MCT6 25031099 Ki = 2560 nM T89034 C5PO7A 25031100 Ki = 3300 nM T89034 CH7Z1K 25031101 Ki = 2900 nM T89034 CEW9X2 25031102 Ki = 2800 nM T89034 C9NC4S 25031541 Ki = 3300 nM T89034 CK5R8Q 25032200 Ki = 1200 nM T89034 CG8HY2 25032202 Ki = 1300 nM T89034 CH76XK 25032204 Ki = 13400 nM T89034 C56GUK 25079268 Ki = 120 nM T89034 CG76TR 25181493 Ki = 120 nM T89034 CKM7Y8 25269170 Ki > 20000 nM T89034 CS5J2O 28742032 Ki > 400000 nM T89034 C54UVP 43165100 Ki = 2511886.43 nM T89034 CPX15D 44188281 IC50 = 0.81 nM T89034 C9OMR4 44264598 Ki > 200000 nM T89034 C9RND0 44264660 Ki > 200000 nM T89034 CHB21I 44265055 IC50 = 500 nM T89034 CVU1T9 44277085 IC50 > 2500 nM T89034 C8Y9JZ 44284991 Ki = 17 nM T89034 CMZ71H 44284992 Ki = 2.9 nM T89034 C5NU9L 44285118 Ki = 24 nM T89034 CU9G2F 44285211 Ki = 5.5 nM T89034 C0FPN1 44285253 Ki = 12 nM T89034 C9N1ZL 44285281 Ki = 4.5 nM T89034 C5PX3O 44285312 Ki = 3 nM T89034 C9LRW8 44285352 Ki = 13 nM T89034 CQ82ZW 44286426 IC50 > 2500 nM T89034 COPR02 44286428 IC50 > 2500 nM T89034 CS5U7F 44286453 IC50 > 2500 nM T89034 C0DG5R 44287043 Ki = 240000 nM T89034 C3QD4W 44287797 Ki > 200000 nM T89034 C5W7SA 44287798 Ki > 200000 nM T89034 C02ARM 44287937 Ki > 200000 nM T89034 CP90NM 44288029 Ki > 200000 nM T89034 CQ7BY9 44289132 Ki > 1000000 nM T89034 CWR03N 44289153 Ki > 1000000 nM T89034 CBU7X1 44289180 Ki > 1000000 nM T89034 C0YV7U 44289263 Ki > 1000000 nM T89034 C1Q7KW 44289264 Ki > 1000000 nM T89034 CD1TP0 44289295 Ki > 1000000 nM T89034 C75NCO 44289296 Ki = 293000 nM T89034 CWZL84 44289297 Ki > 1000000 nM T89034 CUQ35M 44289336 Ki = 279000 nM T89034 CONY81 44289354 Ki = 320000 nM T89034 CZRH12 44290033 IC50 > 11000 nM T89034 CUY95P 44290108 IC50 > 11000 nM T89034 C8APX2 44290947 Ki = 140 nM T89034 CYA94B 44294210 Ki = 2930 nM T89034 C0O2PG 44295723 Ki = 3000 nM T89034 C8AY9O 44296035 Ki = 32000 nM T89034 CQ51FN 44296074 Ki = 10000 nM T89034 C3DG0L 44296128 Ki = 1500 nM T89034 CPF86Z 44296129 Ki = 8800 nM T89034 C38SDX 44296130 Ki = 21000 nM T89034 C1WU8B 44296135 Ki = 2200 nM T89034 C9LGN2 44297867 Ki < 232500 nM T89034 CPM76K 44298377 Ki = 278500 nM T89034 CJU7B0 44298507 Ki = 42500 nM T89034 CRS39A 44298525 Ki = 218000 nM T89034 CQLA16 44303733 Ki > 75000 nM T89034 C5RZL0 44303743 Ki = 650 nM T89034 C16GOI 44303778 Ki = 27000 nM T89034 CN6V9A 44303803 Ki = 6000 nM T89034 CB38WA 44303805 Ki = 4000 nM T89034 CL0U1A 44303806 Ki = 18000 nM T89034 CE0R9A 44303824 Ki > 75000 nM T89034 C5YF7O 44303839 Ki > 75000 nM T89034 C3HXW6 44303858 Ki = 100 nM T89034 CYW9S8 44303912 Ki = 75000 nM T89034 CIQZ37 44303925 Ki > 75000 nM T89034 CJN72A 44303933 Ki = 650 nM T89034 CXCY31 44303935 Ki > 75000 nM T89034 CR4V0L 44304084 Ki > 75000 nM T89034 CG37DH 44304086 Ki > 75000 nM T89034 C7UJH1 44304087 Ki > 75000 nM T89034 CG0R8N 44304097 Ki = 55000 nM T89034 CJ80KE 44304098 Ki > 75000 nM T89034 CG8TI6 44304099 Ki > 75000 nM T89034 C9W8QC 44304100 Ki > 75000 nM T89034 CE31BF 44304104 Ki = 283000 nM T89034 C83YIU 44304139 Ki = 205000 nM T89034 CTOD17 44310306 IC50 = 10000 nM T89034 CMG13A 44310471 IC50 = 74000 nM T89034 C1VKS9 44310574 IC50 = 2500 nM T89034 C1KLY5 44310587 IC50 = 230 nM T89034 C8CJ6O 44310588 IC50 = 740 nM T89034 CK35GH 44310714 IC50 = 460 nM T89034 CNK8W1 44310877 IC50 = 32000 nM T89034 C3X7VO 44313132 IC50 = 8300 nM T89034 CU8S5P 44313405 IC50 = 20000 nM T89034 CIQ1L7 44313498 IC50 = 12200 nM T89034 CF1S3C 44313499 IC50 = 6400 nM T89034 C0G3WT 44313500 IC50 = 25000 nM T89034 CFXW28 44314002 IC50 > 2500 nM T89034 CM10DN 44314053 IC50 = 1200 nM T89034 CCK1W8 44314117 IC50 > 2500 nM T89034 CT1X8J 44314118 IC50 > 2500 nM T89034 CE6B9A 44314318 IC50 > 2500 nM T89034 C4Q9ZF 44315391 Ki > 1000000 nM T89034 C87MBQ 44315392 Ki > 1000000 nM T89034 C5CIL6 44315449 Ki = 576000 nM T89034 C2QOP6 44315450 Ki = 155000 nM T89034 C5WI0G 44315604 Ki > 1000000 nM T89034 CDW83E 44315605 Ki > 1000000 nM T89034 CIBE78 44315607 Ki = 769000 nM T89034 CZ3CY0 44315608 Ki = 214000 nM T89034 C07NBY 44315609 Ki > 1000000 nM T89034 C8DQ5R 44315610 Ki > 1000000 nM T89034 C0Z7PI 44315635 Ki > 1000000 nM T89034 CJ5I9T 44315636 Ki > 1000000 nM T89034 C71UBD 44315637 Ki > 1000000 nM T89034 C8UAJ1 44315641 Ki > 1000000 nM T89034 CH7M1F 44315642 Ki > 1000000 nM T89034 C0EG4V 44315643 Ki > 1000000 nM T89034 C8MU4G 44315644 Ki > 1000000 nM T89034 C2U5HM 44315664 Ki = 700000 nM T89034 CPT78A 44315674 Ki > 1000000 nM T89034 CEO18C 44315675 Ki > 1000000 nM T89034 C25DGE 44315677 Ki > 1000000 nM T89034 C45PHT 44315678 Ki > 1000000 nM T89034 C5QUO9 44315743 Ki > 1000000 nM T89034 CA8L4R 44315744 Ki > 1000000 nM T89034 CPV7S5 44315758 Ki > 1000000 nM T89034 CRVN48 44315788 Ki > 1000000 nM T89034 C1QEV6 44315805 Ki > 1000000 nM T89034 CB7Q2W 44315826 Ki > 1000000 nM T89034 CPH5U7 44315831 Ki > 1000000 nM T89034 CG3VB1 44315832 Ki = 316000 nM T89034 CZ8RS4 44315843 Ki > 1000000 nM T89034 CUGF09 44315844 Ki > 1000000 nM T89034 CX20QR 44315845 Ki > 1000000 nM T89034 C4KF3H 44315846 Ki > 1000000 nM T89034 CCXE57 44315848 Ki > 1000000 nM T89034 C0IVD5 44315849 Ki > 1000000 nM T89034 CU74AZ 44315850 Ki > 1000000 nM T89034 C9QO7H 44315851 Ki > 1000000 nM T89034 CF4I7B 44315852 Ki > 1000000 nM T89034 CS6C5I 44315912 Ki > 1000000 nM T89034 CF48NZ 44315913 Ki > 1000000 nM T89034 C6O5ZT 44315914 Ki = 570000 nM T89034 C8VZ4J 44315915 Ki > 1000000 nM T89034 CZ6K5W 44316015 Ki > 1000000 nM T89034 CUL40O 44316026 Ki > 1000000 nM T89034 CAJ97K 44316048 Ki = 83000 nM T89034 CQ52SH 44316049 Ki > 1000000 nM T89034 C1MRI0 44316050 Ki > 230000 nM T89034 CV38TK 44316051 Ki > 1000000 nM T89034 CKWY45 44316065 Ki > 1000000 nM T89034 CKN8C1 44316486 IC50 > 10000 nM T89034 CK58VB 44318182 IC50 = 271 nM T89034 CEZ84L 44320397 IC50 > 2500 nM T89034 CSK62O 44320493 IC50 > 2500 nM T89034 CYT2Q4 44320495 IC50 > 2500 nM T89034 CG36WH 44320752 IC50 > 2500 nM T89034 CQ64CD 44320839 IC50 > 2500 nM T89034 CK1EZ2 44320862 IC50 > 2500 nM T89034 C7AMH4 44320876 IC50 > 2500 nM T89034 C26KJP 44330423 Ki = 250 nM T89034 C5W1DZ 44330605 IC50 = 141000 nM T89034 C6B0DP 44330620 IC50 = 11000 nM T89034 CW1XE9 44330628 Ki = 230 nM T89034 C1Z5FA 44330631 Ki = 460 nM T89034 CK8FJ6 44330632 Ki > 10000 nM T89034 CS1V3W 44330665 Ki = 250 nM T89034 CQX7A3 44330666 Ki = 14000 nM T89034 CWV7X5 44330835 Ki = 160 nM T89034 C98KLH 44330847 Ki = 140 nM T89034 CSM3B6 44330879 IC50 = 18100 nM T89034 CE69GW 44331194 IC50 = 77900 nM T89034 CN08YB 44331576 Ki = 65600 nM T89034 C98RIJ 44331596 Ki = 43000 nM T89034 CLZ0I6 44331643 Ki > 700000 nM T89034 C58VKT 44331672 Ki > 200000 nM T89034 CKB3M5 44331988 Ki > 1000000 nM T89034 CV6R7F 44331989 Ki > 1000000 nM T89034 C5E7JD 44331991 Ki ~ 200000 nM T89034 CMI8V5 44332049 Ki = 100000 nM T89034 C81IWF 44332152 Ki = 520000 nM T89034 CQHE08 44333168 EC50 = 7650 nM T89034 CNGD56 44333258 EC50 = 2350 nM T89034 C7Y8IG 44334488 Ki = 38 nM T89034 CHL01I 44334805 Ki = 190 nM T89034 C8BKP0 44335014 IC50 = 1500 nM T89034 CE5AZ8 44335512 Ki = 14000 nM T89034 CRT4G3 44335601 Ki = 14000 nM T89034 C7Z9WL 44335624 Ki = 10300 nM T89034 C7TZK3 44335675 Ki = 6100 nM T89034 CS7C2D 44335867 Ki = 6300 nM T89034 C3TVZ2 44335880 Ki = 42000 nM T89034 CHWY63 44336861 Ki = 3000 nM T89034 C0YO9D 44336901 Ki = 6600 nM T89034 C4SE8Q 44336925 Ki = 1800 nM T89034 CYC7S4 44336980 Ki = 1000 nM T89034 CY45FN 44336995 Ki = 21000 nM T89034 C2V8OP 44336996 Ki = 1000 nM T89034 C0DIH9 44336997 Ki = 1500 nM T89034 C73QCK 44337001 Ki = 12000 nM T89034 C5OEX1 44337004 Ki = 3200 nM T89034 C2S4HW 44337018 Ki = 2800 nM T89034 C3W2DF 44337028 Ki = 4500 nM T89034 CR2C7L 44337052 Ki = 2600 nM T89034 C7A3ZN 44337099 Ki = 7100 nM T89034 CO7FI5 44337101 Ki = 9600 nM T89034 C18AZH 44337119 Ki = 2500 nM T89034 C61CGV 44337884 IC50 = 55 nM T89034 C4EFA8 44337894 IC50 = 180 nM T89034 C0HP3T 44337899 IC50 = 400000 nM T89034 CH0K1J 44337917 IC50 = 130 nM T89034 CG6T9S 44337925 IC50 = 41000 nM T89034 CA10BE 44337935 IC50 = 18000 nM T89034 C4ATV2 44337945 IC50 = 620 nM T89034 C2AN5G 44337986 IC50 = 31000 nM T89034 CFH80Q 44337989 IC50 = 15000 nM T89034 CTD5Q8 44338012 IC50 = 21000 nM T89034 C5OVP7 44338032 IC50 > 10000 nM T89034 CI8U6O 44338109 IC50 = 2710 nM T89034 C9WR3T 44338140 IC50 > 2500 nM T89034 CQ37SV 44339192 Ki = 47500 nM T89034 C8JQA9 44339233 Ki = 237800 nM T89034 CU52DY 44339260 Ki = 24000 nM T89034 C3XI4S 44339270 Ki = 47500 nM T89034 CU20ZI 44339271 Ki = 12000 nM T89034 C98MCJ 44339277 Ki = 50800 nM T89034 C7CAT2 44339282 Ki = 131400 nM T89034 CX3B5S 44339419 Ki = 4750 nM T89034 CBU40W 44339439 Ki = 3200 nM T89034 CKA1T3 44341287 IC50 = 315 nM T89034 CZ9BF5 44341288 IC50 = 923 nM T89034 C4XEK1 44341417 IC50 = 14.8 nM T89034 CC0Z8V 44343581 IC50 = 367 nM T89034 CW76HT 44343582 IC50 = 673 nM T89034 CD0TW8 44343615 IC50 = 521 nM T89034 CAIZ35 44343800 IC50 = 1140 nM T89034 C0W6EI 44343845 IC50 = 1480 nM T89034 C46IGW 44343852 IC50 > 2500 nM T89034 C5H3NY 44343853 IC50 > 2500 nM T89034 C40EHX 44343858 IC50 = 1440 nM T89034 C91PVF 44343859 IC50 = 700 nM T89034 C4MS5Q 44343972 IC50 > 2500 nM T89034 C3ZI7A 44343993 IC50 = 2030 nM T89034 CMEI89 44343994 IC50 = 1140 nM T89034 CEA17Z 44344039 IC50 = 3270 nM T89034 CUO74X 44344054 IC50 = 1060 nM T89034 C60GZW 44344100 IC50 = 250 nM T89034 CREZ48 44344153 IC50 = 2500 nM T89034 CAY34C 44347478 Ki = 744000 nM T89034 CT0QN1 44347480 Ki > 1000000 nM T89034 C1UN9I 44347534 Ki > 1000000 nM T89034 C0V2FL 44347624 Ki = 572000 nM T89034 CX9MJ6 44356715 Ki = 1190 nM T89034 C81XMY 44358802 IC50 = 8100 nM T89034 CPX09V 44358866 IC50 = 740000 nM T89034 CSNJ26 44358867 IC50 = 850000 nM T89034 CL0U6H 44358868 IC50 = 11000 nM T89034 CUE9P4 44359039 IC50 = 340 nM T89034 C2NQC0 44359053 IC50 = 360 nM T89034 C2P6RJ 44364043 Ki = 50000 nM T89034 C06RPS 44364101 Ki = 10000 nM T89034 CN46VL 44364123 Ki = 10000 nM T89034 CYK89L 44364205 Ki = 10000 nM T89034 CP7K4W 44364302 Ki = 25000 nM T89034 C4LH6Q 44364310 Ki = 14000 nM T89034 CB85LE 44364311 Ki = 50000 nM T89034 CDE32K 44364319 Ki = 25000 nM T89034 CTC3O5 44364320 Ki = 25000 nM T89034 CSI3V9 44364329 Ki = 25000 nM T89034 CUM70S 44364371 Ki = 26000 nM T89034 C9Z7JD 44364382 Ki = 44000 nM T89034 CTB86G 44364486 Ki = 52000 nM T89034 C1ELX6 44364487 Ki = 50000 nM T89034 CS2D1R 44364505 Ki = 40000 nM T89034 CQE3K8 44364506 Ki = 45000 nM T89034 C39FZP 44372663 Ki = 140000 nM T89034 C9I0BE 44372667 Ki = 2400 nM T89034 CQLA75 44372683 Ki = 75000 nM T89034 CKFN05 44372724 Ki > 1000000 nM T89034 CTD36H 44372738 Ki > 1000000 nM T89034 CI6MQ5 44372778 Ki = 43000 nM T89034 CFH41R 44372839 Ki = 17000 nM T89034 C9COY7 44372840 Ki > 1000000 nM T89034 C34AWY 44372863 Ki = 160000 nM T89034 CZE15A 44372864 Ki = 32000 nM T89034 C7X5BE 44372865 Ki = 150 nM T89034 C2E6TP 44372889 Ki = 59000 nM T89034 C36XWM 44372903 Ki = 150 nM T89034 C34XTM 44375987 IC50 = 309 nM T89034 CD0W7C 44376100 IC50 = 10700 nM T89034 C0Y8QD 44376252 IC50 = 1880 nM T89034 C5R2PM 44376328 IC50 = 1300 nM T89034 C5VDG0 44376417 IC50 = 10 nM T89034 CG64YQ 44376426 IC50 = 121 nM T89034 CI2GS0 44377287 IC50 = 965 nM T89034 C7W2GD 44377304 IC50 = 894 nM T89034 CP0V6X 44377320 IC50 = 387 nM T89034 C4KSG5 44377322 IC50 > 2500 nM T89034 CH1NM4 44377327 IC50 > 2500 nM T89034 CTP28F 44377331 IC50 = 678 nM T89034 C30VGP 44377425 IC50 = 1190 nM T89034 CT0G2D 44377544 IC50 = 1440 nM T89034 CK6I3F 44377546 IC50 = 872 nM T89034 CNUL43 44377548 IC50 = 231 nM T89034 CZBJ51 44377550 IC50 = 2500 nM T89034 CHU5T4 44377558 IC50 = 2500 nM T89034 CD36KV 44380417 Ki = 490 nM T89034 CJ6M5B 44382389 IC50 > 2500 nM T89034 CTF4N6 44382391 IC50 = 250 nM T89034 CAI65F 44382441 IC50 > 2500 nM T89034 C6LH5V 44383081 IC50 > 2500 nM T89034 C9SD3E 44383242 Ki > 7300 nM T89034 C5PW9E 44383425 IC50 > 2500 nM T89034 C43KTU 44383519 Ki > 7300 nM T89034 CNBG48 44383542 IC50 > 2500 nM T89034 C2IX5U 44383543 IC50 > 2500 nM T89034 CQ05YV 44384709 IC50 < 1000 nM T89034 CG7LT1 44385488 IC50 > 11000 nM T89034 C94GZU 44385541 IC50 > 11000 nM T89034 C3T9XK 44385607 IC50 > 11000 nM T89034 CKY0P4 44385611 IC50 > 11000 nM T89034 CUS20V 44385673 IC50 > 11000 nM T89034 CZ8XL6 44385679 IC50 > 11000 nM T89034 COQH07 44385725 IC50 = 1170 nM T89034 CL5BA4 44385729 IC50 > 11000 nM T89034 C3DSN7 44385768 IC50 > 11000 nM T89034 C8USN9 44385769 IC50 > 11000 nM T89034 CX9W5Z 44385770 IC50 = 275 nM T89034 C2E8DS 44385771 IC50 > 11000 nM T89034 C2VFC6 44385772 IC50 > 11000 nM T89034 CN8V0W 44385779 IC50 > 11000 nM T89034 C7MXA5 44385833 IC50 = 904 nM T89034 CBEA65 44385842 IC50 > 11000 nM T89034 CC9M7E 44385869 IC50 > 11000 nM T89034 C8WK4A 44385891 IC50 > 11000 nM T89034 C3D2CL 44385935 IC50 > 11000 nM T89034 CW08OY 44385998 IC50 > 11000 nM T89034 C8F2RG 44386052 IC50 = 125 nM T89034 CV6KG4 44386059 IC50 > 11000 nM T89034 CGU69V 44386179 IC50 > 11000 nM T89034 CS65LH 44386185 IC50 > 11000 nM T89034 CU0P5T 44386242 IC50 > 11000 nM T89034 CU9J0D 44386250 IC50 > 11000 nM T89034 C9G7QW 44386322 IC50 > 11000 nM T89034 C31CUG 44386326 IC50 > 11000 nM T89034 C52MCK 44386366 IC50 = 482 nM T89034 C2WCE4 44386371 IC50 > 11000 nM T89034 C52POK 44386417 IC50 > 11000 nM T89034 CRX1I9 44386418 IC50 > 11000 nM T89034 CBG1U6 44386478 IC50 = 699 nM T89034 CIBD76 44386484 IC50 > 11000 nM T89034 C8ME4O 44386493 IC50 > 11000 nM T89034 CD4AH3 44386540 IC50 > 11000 nM T89034 CHAO48 44386542 IC50 > 11000 nM T89034 CLNO15 44386637 IC50 > 11000 nM T89034 C81IMH 44386642 IC50 > 11000 nM T89034 CWTU45 44386804 IC50 > 2500 nM T89034 C4JB0M 44386841 IC50 > 11000 nM T89034 CA0W2K 44386893 IC50 > 2500 nM T89034 C5MR1F 44386934 IC50 > 11000 nM T89034 CA45DZ 44387044 IC50 > 11000 nM T89034 C39LUW 44387104 IC50 > 11000 nM T89034 C2QD1K 44387206 IC50 > 11000 nM T89034 CG52IR 44391923 Ki = 23000 nM T89034 CAY27D 44392382 Ki = 1480 nM T89034 C2SQ1C 44392401 Ki = 1015 nM T89034 C4VKE9 44392403 Ki = 277 nM T89034 CYL52J 44392413 Ki = 243 nM T89034 CN8CJ3 44392416 Ki = 239 nM T89034 CE42KB 44392423 Ki = 570 nM T89034 CORK28 44392427 Ki = 2454 nM T89034 C78QJO 44394249 Ki > 50000 nM T89034 CQRB69 44394250 Ki > 50000 nM T89034 CB0N5T 44400527 Ki = 78200 nM T89034 CNRA17 44404044 IC50 = 6600 nM T89034 CJ8E3S 44404045 IC50 = 13500 nM T89034 C4R2GU 44404046 IC50 = 3200 nM T89034 CSQ76C 44404047 IC50 = 3300 nM T89034 C7JT3R 44404048 IC50 = 3600 nM T89034 CTS5W9 44404049 IC50 = 2700 nM T89034 CY6NZ8 44404050 IC50 = 14100 nM T89034 CP67EA 44411094 IC50 = 1470 nM T89034 CM8OZ0 44411137 IC50 > 20000 nM T89034 CB1G3D 44412151 Ki = 2900 nM T89034 CC2Z1K 44412258 Ki = 4030 nM T89034 CLQ54S 44412280 Ki > 100000 nM T89034 C3BX5Y 44412781 Ki = 910 nM T89034 CF5XO4 44413343 Ki = 1800 nM T89034 CTD42X 44413355 Ki = 2800 nM T89034 C9KQM2 44413356 Ki = 3100 nM T89034 CQDX92 44413619 Ki = 800 nM T89034 CPN1S0 44416248 IC50 = 5000 nM T89034 CVO5Q1 44432538 Ki > 22000 nM T89034 CR16BF 44434808 Ki > 22000 nM T89034 CQIX73 44434809 Ki > 22000 nM T89034 C5R8HJ 44434815 Ki > 22000 nM T89034 COG34X 44434818 Ki > 22000 nM T89034 C9T1DP 44434835 Ki > 22000 nM T89034 C30CFX 44436704 IC50 = 30000 nM T89034 CB86HU 44453827 IC50 = 36 nM T89034 CH4IG1 44459090 Ki > 500000 nM T89034 CV5TB1 44459377 Ki > 500000 nM T89034 CVBZ10 44459392 Ki = 34000 nM T89034 CGS82Z 44459487 Ki > 500000 nM T89034 C95MDP 44459488 Ki > 500000 nM T89034 CJ16HT 44459496 Ki > 500000 nM T89034 CZC3P9 44459497 Ki > 500000 nM T89034 CWB04E 44462312 IC50 > 2500 nM T89034 CEW6G1 44569299 Ki = 28 nM T89034 C9JNT3 44569300 Ki = 210 nM T89034 C9XE7Q 44569301 Ki = 16000 nM T89034 CZI8D7 44569333 Ki = 64800 nM T89034 CR4CP6 44569359 Ki = 776 nM T89034 C9JF7W 44569667 Ki = 200 nM T89034 C61IJB 44569732 Ki = 460 nM T89034 CR36MB 44569733 Ki = 2600 nM T89034 CE25UL 44569767 Ki = 3500 nM T89034 C0CZ4I 44569768 Ki = 2100 nM T89034 CIR4M0 44569769 Ki = 550 nM T89034 C02SHD 44569811 Ki = 85 nM T89034 CG3LE9 44569812 Ki = 334 nM T89034 CCU7V0 44569813 Ki = 183 nM T89034 C8BR6E 44569843 Ki = 150 nM T89034 C7Q9BH 44569844 Ki = 80 nM T89034 CZ35OW 44569845 Ki = 230 nM T89034 CHV9C1 44569846 Ki = 214 nM T89034 C5JQ4W 44569889 Ki = 110 nM T89034 CE1O4I 44569890 Ki = 1000 nM T89034 C4JU7I 44569891 Ki = 380 nM T89034 CGS83Z 44569892 Ki = 230 nM T89034 C4BN3H 44573109 Ki = 1600 nM T89034 COR57Y 44573272 Ki = 6200 nM T89034 C6DX3Y 44573273 Ki = 2800 nM T89034 CM2R1P 44573274 Ki = 3600 nM T89034 CSP1I0 44573310 Ki = 2500 nM T89034 C6EG9V 44573311 Ki = 9400 nM T89034 CYV3X2 44573378 Ki = 4500 nM T89034 CWUA41 44573379 Ki = 4900 nM T89034 CYA64G 44573380 Ki = 69400 nM T89034 CLG42S 44573428 Ki = 79000 nM T89034 CI5C1F 44592560 IC50 = 0.308 nM T89034 CNIX06 44592593 IC50 = 0.358 nM T89034 CZJ7C6 44592617 IC50 > 5 nM T89034 C1A8YB 44592658 IC50 > 5 nM T89034 CC65UK 44592729 IC50 = 0.163 nM T89034 CKC2Q8 44592831 IC50 = 0.06 nM T89034 CY2IM4 44592833 IC50 = 0.242 nM T89034 CW72YN 44592864 IC50 = 0.457 nM T89034 CD4G2B 44592865 IC50 = 0.554 nM T89034 CDLY78 44592888 IC50 = 0.656 nM T89034 C1PLT5 44592978 IC50 > 5 nM T89034 CVS21G 44592979 IC50 = 1 nM T89034 C4M0KI 44593006 IC50 = 0.07 nM T89034 C9PCO6 44593008 IC50 = 0.684 nM T89034 C8XT1U 44626341 IC50 = 1900 nM T89034 C7JP5Q 44626343 IC50 = 5000 nM T89034 CDG17C 44626344 IC50 = 5500 nM T89034 C6I0TN 44626345 IC50 = 3000 nM T89034 C2PVE0 45103523 Ki > 26000 nM T89034 CGN14R 45103723 Ki > 26000 nM T89034 CEXO72 45261244 IC50 = 71000 nM T89034 CGXD19 45485586 IC50 = 2100 nM T89034 C9OZ8H 45485587 IC50 = 6500 nM T89034 C0H5ST 45485592 IC50 = 9400 nM T89034 CPT2Y1 45485611 IC50 = 11000 nM T89034 C27HKO 45485622 IC50 = 5000 nM T89034 CF39BN 45485632 IC50 = 2700 nM T89034 C3HKP7 45485641 IC50 = 3600 nM T89034 C62BQW 45485647 IC50 = 8600 nM T89034 C7UK5D 45485655 IC50 = 2800 nM T89034 CHT06J 45485667 IC50 = 2900 nM T89034 C76CDZ 45485668 IC50 = 2100 nM T89034 CGX93B 45485669 IC50 = 4400 nM T89034 C0R4EB 45485670 IC50 = 6300 nM T89034 CI5EJ4 45485671 IC50 = 21000 nM T89034 CJ73BT 45486346 Ki = 97000 nM T89034 C9ETC4 45486354 Ki > 1000000 nM T89034 CCG5U1 46196561 Ki > 60000 nM T89034 C4YAJ7 46228924 IC50 > 100000 nM T89034 CF58MH 46883093 IC50 = 0.1 ug.mL-1 T89034 C4OCL0 46883094 IC50 = 0.4 ug.mL-1 T89034 CNVR31 46905372 IC50 = 37000 nM T89034 CMD0O1 46937699 IC50 = 770 nM T89034 C6WX5V 46937701 IC50 = 450 nM T89034 C9GQZ7 46937704 IC50 = 1260 nM T89034 C7PBI9 46938035 IC50 = 580 nM T89034 C4RAB3 46938036 IC50 = 169000 nM T89034 CU90MG 46938037 IC50 = 280 nM T89034 CC9U7X 46938038 IC50 = 150000 nM T89034 C95ESD 46938041 IC50 = 1020 nM T89034 CX2U5I 46938097 IC50 = 390 nM T89034 C47QBL 46938101 IC50 = 1500 nM T89034 C7O5IV 46938160 IC50 = 1060 nM T89034 CS8FY6 49820655 Ki = 1205 nM T89034 CL8UV3 49820969 Ki = 8 nM T89034 CU1DK9 49835415 Ki = 63 nM T89034 C0OQ8N 49835557 Ki = 17.5 nM T89034 CLOY62 49864459 Ki > 33000 nM T89034 CR8JK9 49864483 Ki > 33000 nM T89034 CA86OS 53317375 Ki = 1000000 nM T89034 C7QEI1 53321291 Ki = 1000000 nM T89034 CFOI53 53322612 Ki = 400000 nM T89034 CWA7B3 53323948 Ki = 1000000 nM T89034 CO6TG4 53325236 Ki = 1000000 nM T89034 CO0R2M 53325237 Ki = 110000 nM T89034 CA6GQ5 53341037 Ki > 15200 nM T89034 CIKQ81 53345652 Ki = 0.25 nM T89034 CXWS90 53345968 Ki = 0.6 nM T89034 C76GSI 53346181 Ki = 3 nM T89034 CB08CW 53379392 Ki = 23130 nM T89034 CV60BK 53488415 Ki = 15780 nM T89034 C17MSO 56640092 Ki = 6.9 nM T89034 CGP7Y6 56640160 Ki = 4.1 nM T89034 C30AJK 56640226 Ki = 1.1 nM T89034 C8U4OD 56649692 IC50 > 1000000 nM T89034 CA32CM 56659850 Ki = 590 nM T89034 CKO4M6 56663319 Ki = 2110 nM T89034 CCM80T 56670171 Ki = 1520 nM T89034 CGM2J4 56673694 Ki = 2810 nM T89034 C4T6NO 56673695 Ki = 161 nM T89034 C1TH3W 56677006 Ki = 114 nM T89034 CY34VE 56677007 Ki = 3030 nM T89034 C72IHP 56680339 Ki = 1160 nM T89034 CH1EI8 56954620 Ki = 431 nM T89034 C4EHU8 56954732 Ki = 9.4 nM T89034 C5C8XO 56954733 Ki = 9 nM T89034 CST4F0 56954834 Ki = 1.1 nM T89034 CRK92A 56954952 Ki = 2.2 nM T89034 CLU95A 57325502 IC50 > 62000 nM T89034 CTJ5Z3 57390228 IC50 = 290000 nM T89034 CLY4C9 57390236 IC50 = 220000 nM T89034 CV42AN 57390824 IC50 = 20000 nM T89034 C1GIV7 57390825 IC50 = 31000 nM T89034 CM7FT5 57390879 IC50 > 125000 nM T89034 C5Q7IU 57393748 IC50 = 140000 nM T89034 CEO1L3 57393799 IC50 = 220000 nM T89034 CXV4U9 57394359 IC50 = 6300 nM T89034 CR9HP7 57397305 IC50 = 78000 nM T89034 C4CQ9K 57397312 IC50 = 370000 nM T89034 CIC2U6 57397927 IC50 = 12000 nM T89034 C6QJ7Y 57400705 IC50 = 590000 nM T89034 CXZ3D0 57400764 IC50 = 570000 nM T89034 CKV6R8 57401327 IC50 = 6500 nM T89034 C45RAM 57402478 IC50 = 240000 nM T89034 CES6D2 57403083 IC50 = 4000 nM T89034 C3RZ8G 57404502 IC50 > 250000 nM T89034 CVWP51 57404503 IC50 > 250000 nM T89034 C9XW1C 57842830 Ki > 10000 nM T89034 C60HCV 57976401 Ki > 15200 nM T89034 CHB27Y 57976410 Ki = 12540 nM T89034 CM8UJ7 57976444 Ki > 24000 nM T89034 CQ71KE 57976446 Ki > 41000 nM T89034 CPW2H7 59315536 Ki > 10000 nM T89034 CE5A7B 60162406 Ki = 0.68 nM T89034 CE54UJ 66732202 IC50 = 360 nM T89034 CWOD93 66744646 Ki > 14200 nM T89034 C6LD2R 66818559 Ki = 22 nM T89034 C6CP8D 66818568 Ki = 13 nM T89034 C05LHZ 66818575 Ki = 2395 nM T89034 C9GM3F 66818639 Ki = 13 nM T89034 C4U7SZ 66818677 Ki = 2410 nM T89034 C6Q8FO 66818744 Ki = 2160 nM T89034 CR94HZ 66818781 Ki = 2630 nM T89034 CP18VA 66818813 Ki = 3610 nM T89034 CF4PT6 66818819 Ki = 8 nM T89034 CYB76J 66818882 Ki = 8 nM T89034 CGI6B3 66819113 Ki = 2590 nM T89034 C4JV1L 66820910 Ki = 3855 nM T89034 CKWQ82 67155200 Ki = 29000 nM T89034 C0SDB3 68020667 Ki = 0.57 nM T89034 CGA3T2 68789018 Ki = 10 nM T89034 CC0J3V 68790735 Ki = 16 nM T89034 CPY6J2 69496521 IC50 = 5100 nM T89034 CPO6Z9 69496614 IC50 = 3325 nM T89034 C1DUV4 69496716 IC50 > 30000 nM T89034 C6YW5E 69496717 IC50 = 1900 nM T89034 CUG9Z7 69496724 IC50 = 5450 nM T89034 CR59OP 69496744 IC50 = 1850 nM T89034 CX97VL 69496820 IC50 = 1330 nM T89034 CD5ZW0 69496838 IC50 = 5400 nM T89034 CA49UK 69520512 Ki > 19000 nM T89034 C6AU1R 70252985 Ki = 38100 nM T89034 CTO5I6 70253788 Ki > 53400 nM T89034 C8A7ZJ 70306716 Ki = 2.2 nM T89034 CL4RK8 70683232 IC50 > 250000 nM T89034 C4IFW3 70683249 Ki = 0.81 nM T89034 C0G1ZN 70685354 Ki = 530 nM T89034 CN38UY 70687492 Ki = 2.5 nM T89034 CX0VK6 70689516 IC50 > 250000 nM T89034 C2UOG4 70693724 IC50 > 150000 nM T89034 CWEP17 70693749 Ki = 3.08 nM T89034 CE27BR 70695842 IC50 > 250000 nM T89034 C9EL3C 71260387 Ki > 15200 nM T89034 C45SHM 71451304 Ki > 20000 nM T89034 C0XV2L 71455698 IC50 = 99000 nM T89034 C1UOK5 71458276 EC50 = 4900 nM T89034 CJPF90 71548883 Ki > 25000 nM T89034 C30ZKJ 71561420 Ki = 0.2 nM T89034 CH32TL 71561557 Ki = 0.52 nM T89034 C8RW7E 71562631 Ki = 7 nM T89034 C4UHB2 71562760 Ki = 9 nM T89034 C0EM6D 71562761 Ki = 5.1 nM T89034 CNS21T 71562882 Ki = 4 nM T89034 C3SBE2 71562883 Ki = 1.32 nM T89034 C2NY0B 71563006 Ki = 1.15 nM T89034 CG46AZ 71563007 Ki = 1.62 nM T89034 C2O4SB 71563124 Ki = 0.76 nM T89034 C4CT8O 71563125 Ki = 1.71 nM T89034 C78DJQ 71711730 IC50 < 10000 nM T89034 CC3ZD4 71716372 Ki = 14200 nM T89034 C5ET1Z 71716373 Ki = 8300 nM T89034 CD53RA 71716975 Ki > 120000 nM T89034 CSP5T2 71716976 Ki = 8300 nM T89034 CD12XQ 71716977 Ki > 120000 nM T89034 CR9KP1 71717597 Ki > 120000 nM T89034 CHM12E 71718213 Ki = 3300 nM T89034 CK8VH9 71718214 Ki = 118300 nM T89034 CD8GN0 71718815 Ki = 4300 nM T89034 CBN5O8 71718816 Ki > 120000 nM T89034 C42ODM 71718819 Ki > 120000 nM T89034 CQ3K2V 71719191 Ki = 25 nM T89034 CK73ZJ 71720640 Ki > 120000 nM T89034 CM83VP 72163524 IC50 > 10000 nM T89034 CLI36U 72551247 Ki = 1500 nM T89034 CDQP51 73347119 Ki > 50000 nM T89034 C5AMR2 73348056 IC50 > 100000 nM T89034 CB8RP9 73350124 IC50 = 230 nM T89034 CAJ7O5 73350148 Ki > 1000000 nM T89034 CM3PH8 73350210 Ki > 50000 nM T89034 CL8EG7 73350757 Ki = 7430 nM T89034 CAW4V2 73353028 Ki = 9000000 nM T89034 C60JSR 73353029 Ki = 50000 nM T89034 C5U9CI 73355715 Ki = 0.01 nM T89034 CL6X7D 76335180 IC50 = 6 ug.mL-1 T89034 C9ASZ2 86302628 IC50 = 14000 nM T89034 CMD5V7 86583041 Ki > 22100 nM T89034 CV7IW5 87167024 Ki = 5 nM T89034 CO6U9I 88582319 Ki = 76600 nM T89034 C3Z6DC 89952799 IC50 = 100000 nM T89034 CJ6CN0 90644019 Ki = 2665 nM T89034 C0G6SP 90644022 Ki = 1530 nM T89034 C1KF8D 90644590 IC50 = 40000 nM T89034 CK0HQ8 90644591 IC50 = 2100 nM T89034 C9A7YX 90655485 IC50 > 1000000 nM T89034 C90UNY 90655486 IC50 = 43000 nM T89034 C75WHK 90655487 IC50 = 180000 nM T89034 CZ1Q2P 90655488 IC50 = 330000 nM T89034 CSG0L5 90655489 IC50 = 260000 nM T89034 C8KX5F 90655490 IC50 = 160000 nM T89034 C9W1CO 90655491 IC50 = 210000 nM T89034 C5WIF7 90655492 IC50 = 220000 nM T89034 C6FE2K 90655493 IC50 = 100000 nM T89034 C2I7SQ 90655494 IC50 = 220000 nM T89034 CXY0I6 90655495 IC50 = 250000 nM T89034 CWL8U1 90655496 IC50 = 400000 nM T89034 CRQ6I4 90655497 IC50 = 130000 nM T89034 CL27GQ 90655498 IC50 = 64000 nM T89034 CLG8M0 90655499 IC50 = 87000 nM T89034 CBK7Y9 90655500 IC50 > 250000 nM T89034 CD7WM6 90655501 IC50 = 99000 nM T89034 CJ7B8Y 90655502 IC50 = 510000 nM T89034 CW6VS9 90655503 IC50 = 170000 nM T89034 CV1NM4 90655504 IC50 = 510000 nM T89034 CKPN23 90655505 IC50 > 250000 nM T89034 CZ8S4C 90655506 IC50 = 960000 nM T89034 CG83WX 90655748 Ki = 15848.93 nM T89034 CK3P6X 91667569 IC50 = 8.6 nM T89034 C65TLW 101862198 Ki > 1000000 nM T89034 C98BXU 117984620 IC50 = 0.8 nM T89034 CH5Z4P 117985339 IC50 = 0.32 nM T89034 CPAC38 117986252 IC50 = 23 nM T89034 C3KB4M 117986600 IC50 = 0.4 nM T89034 CI4KC5 117986603 IC50 = 0.87 nM T89034 CMJ8R1 118601604 Ki = 36 nM T89034 C0GRU4 118718129 Ki = 7.8 nM T89034 CGL2B0 118725262 Ki = 63095.73 nM T89034 CHQ5P7 118987013 Ki > 22100 nM T89034 CUM06Y 122179831 IC50 = 43000 nM T89034 CK89ZG 122179832 IC50 = 26000 nM T89034 CB6C8Y 122179833 IC50 = 29000 nM T89034 CCN75S 122179834 IC50 = 23000 nM T89034 C4A3JB 122179835 IC50 = 130000 nM T89034 C7MJB0 122179836 IC50 = 160000 nM T89034 C81TAC 122179837 IC50 > 200000 nM T89034 C5EN4W 122179838 IC50 > 200000 nM T89034 CTPA56 122179839 IC50 = 100000 nM T89034 C6GO7H 122179840 IC50 > 200000 nM T89034 CBM46S 122179841 IC50 = 25000 nM T89034 CY51OU 122179842 IC50 = 74000 nM T89034 CB8K4S 122179843 IC50 = 56000 nM T89034 C4B0JR 122179844 IC50 > 200000 nM T89034 CP42JE 122192779 Ki = 14300 nM T89034 C43TNZ 122192780 Ki = 17100 nM T89034 C71IOQ 122192783 Ki = 121 nM T89034 CNJH01 122192784 Ki = 549 nM T89034 CR7MG0 122224465 IC50 = 45000 nM T89034 C2V6PQ 122550396 IC50 = 1 nM T89034 C8NR0Y 122550417 IC50 = 2.1 nM T89034 C3W6DG 122551266 IC50 = 0.42 nM T89034 CFD89O 127021019 IC50 = 220 nM T89034 CB9V3Y 127025119 IC50 = 750 nM T89034 C8UHI6 127025120 Ki = 2900 nM T89034 CQHF03 127026968 IC50 = 7700 nM T89034 CKRS95 127026969 IC50 = 11000 nM T89034 CJ6DA9 127028140 IC50 > 10000 nM T89034 CD9KI3 127028141 IC50 > 10000 nM T89034 CPC0M8 127031390 Ki > 22100 nM T89034 C3XD2I 127035151 IC50 = 970 nM T89034 C1BWV2 127035672 Ki = 12500 nM T89034 COG73V 127035809 IC50 = 17000 nM T89034 C07FSI 127035810 IC50 = 1700 nM T89034 C73SHP 127035840 IC50 = 600 nM T89034 CBJ14T 127035841 IC50 = 960 nM T89034 CM34NK 127035842 IC50 = 1500 nM T89034 C6TS0X 127035843 IC50 = 510 nM T89034 C6W4AT 127035844 IC50 = 530 nM T89034 CL6HJ1 127036010 IC50 = 490 nM T89034 CFWR36 127036011 IC50 = 2700 nM T89034 CHQ42U 127036012 IC50 = 1600 nM T89034 CVRY56 127036086 Ki = 10600 nM T89034 C54OHE 127036643 IC50 = 680 nM T89034 CJ0L7S 127036644 IC50 = 860 nM T89034 CN42TJ 127036645 IC50 = 3000 nM T89034 C76FJU 127036847 IC50 = 710 nM T89034 CK40VA 127036848 IC50 = 340 nM T89034 C9B6LT 127037264 Ki = 9800 nM T89034 C60HLK 127037469 Ki > 1000000 nM T89034 C64FQM 127037562 IC50 = 67000 nM T89034 C85ROH 127041472 IC50 > 100000 nM T89034 C8MKE9 127045985 IC50 = 19000 nM T89034 C6T3JF 127045986 IC50 = 28000 nM T89034 CV4TI5 127045987 IC50 = 4900 nM T89034 CK6D1Z 127045988 IC50 = 6700 nM T89034 C3ZP4A 127046388 IC50 = 25000 nM T89034 C8IVS0 127046389 IC50 = 45000 nM T89034 CBL5K4 127046390 IC50 = 19000 nM T89034 C6TYG9 127046555 IC50 = 12000 nM T89034 CHDW47 127046556 IC50 = 11000 nM T89034 C21JMT 127046792 IC50 = 7700 nM T89034 CT2RV6 134130781 IC50 > 1000000 nM T89034 CWV3G6 134131077 IC50 = 9970 nM T89034 CS8FV1 134131084 IC50 > 200000 nM T89034 C92RTL 134131303 IC50 = 21400 nM T89034 CL37SG 134131589 IC50 > 200000 nM T89034 C6HTD5 135393470 IC50 > 10000 nM T89034 C7NA6E 135393474 IC50 > 20000 nM T89034 CD53CZ 135404951 Ki > 7300 nM T89034 C5XA6H 135407717 Ki = 35000 nM T89034 C0OX6T 135407736 Ki = 41000 nM T89034 C61XOA 135427245 Ki = 19000 nM T89034 C8WS4O 135443730 Ki = 60000 nM T89034 CTP5V8 135444609 Ki = 5000 nM T89034 C9KLD3 135455964 Ki = 6200 nM T89034 CJWC64 135462427 Ki = 2350 nM T89034 CXS6B9 135471524 Ki = 7500 nM T89034 C2PFI8 135475618 Ki = 15000 nM T89034 CBE9G0 135490854 Ki = 33000 nM T89034 CMQ6O0 135501618 Ki = 60000 nM T89034 CVA61N 135512760 Ki = 29000 nM T89034 CK97FT 135533257 Ki = 4100 nM T89034 CAD75F 135535997 Ki = 12000 nM T89034 CCH49A 135544551 Ki = 5500 nM T89034 CKLD47 135544579 Ki = 80000 nM T89034 C91UXW 135802775 Ki = 3500 nM T89034 CQD2Z1 135855944 Ki = 3.2 nM T89034 C9G7TE 135995982 Ki = 4200 nM T89034 C6S5OL 136034781 Ki = 47000 nM T89034 CYQ70K 136053621 IC50 > 11000 nM T89034 CN70IU 136092208 Ki = 1600 nM T89034 C5N3KP 136092209 Ki = 1700 nM T89034 C1BUH6 136092210 Ki = 21000 nM T89034 CFQ2C8 136092211 Ki = 3000 nM T89034 CX5R9J 136092212 Ki = 3100 nM T89034 C35PXN 136092213 Ki = 1600 nM T89034 CEXJ30 136092214 Ki = 1800 nM T89034 CS6QH0 136092215 Ki = 1000 nM T89034 CMR7L4 136092216 Ki = 27000 nM T89034 CN0WR7 136092217 Ki = 4200 nM T89034 COCN35 136092218 Ki = 850 nM T89034 CA79JC 136092219 Ki = 1600 nM T89034 CPK6X2 136198635 Ki = 3600 nM T89034 CRJ5S4 136198636 Ki = 7300 nM T89034 C7WE2G 136198637 Ki = 4500 nM T89034 C12UWY 136198638 Ki > 7300 nM T89034 C26ZPI 136264091 IC50 > 250000 nM T89034 C8VJW4 136266885 IC50 > 250000 nM T89034 CC0BI4 136268735 IC50 > 250000 nM T89034 C2JT1W 137632528 IC50 = 116000 nM T89034 CZ9X0E 137634272 IC50 = 47000 nM T89034 CDQ62V 137637214 Ki > 50000 nM T89034 C43ETF 137637257 IC50 = 121000 nM T89034 C3M2QT 137637957 IC50 = 282000 nM T89034 C2K8JV 137639385 Ki > 50000 nM T89034 C50WFO 137642080 IC50 > 1000000 nM T89034 CC7QL4 137642978 IC50 = 14000 nM T89034 C7BQ8O 137644210 IC50 = 34000 nM T89034 C9BEA1 137644608 IC50 = 71000 nM T89034 C6BE7C 137646856 IC50 = 34000 nM T89034 CNO2T8 137647340 IC50 = 3600 nM T89034 CME1B3 137649275 IC50 = 231000 nM T89034 C7WRB2 137652193 IC50 = 73000 nM T89034 CNX46H 137654508 Ki > 50000 nM T89034 CZ1H4R 137655362 Ki > 10000 nM T89034 C47IZA 137655464 IC50 = 76000 nM T89034 CVN59W 137656193 IC50 = 20000 nM T89034 C34UDN 137657165 IC50 = 37000 nM T89034 C0C5JK 137657334 IC50 = 6500 nM T89034 CTUM82 137658421 IC50 = 42000 nM T89034 CO51HN 139030452 IC50 > 20000 nM T89034 CX07YE 139592452 Ki > 15200 nM T89034 C41LXH 145960914 Ki = 140 nM T89034 CE6C0A 145970642 Ki = 4490 nM T89034 CZ1R3B 145982984 Ki = 2.2 nM T89034 C4HLX8 146029523 IC50 > 20000 nM T89034 CH59QO 155510375 Ki = 0.43 nM T89034 CER7V8 155511309 Ki = 0.66 nM T89034 C3U8GK 155511607 IC50 = 0.4 nM T89034 CA81QV 155512709 Ki = 1.2 nM T89034 C2VX3G 155512946 Ki > 15000 nM T89034 CYT20V 155514020 Ki = 0.051 nM T89034 CNM7H8 155514372 IC50 = 20000 nM T89034 CAT98N 155514640 Ki = 270 nM T89034 CG9H4N 155515624 Ki = 66.3 nM T89034 C7ZM4R 155515728 Ki = 3.93 nM T89034 CW3JV1 155516308 Ki = 0.66 nM T89034 CPUG37 155516479 Ki > 19000 nM T89034 CFRS54 155516565 Ki = 3.7 nM T89034 C1ZSV0 155517054 Ki = 75.3 nM T89034 CF96DM 155518671 Ki > 10000 nM T89034 C7DUX3 155520916 Ki = 1500 nM T89034 C4VU1P 155522856 Ki = 1.1 nM T89034 C1JH5P 155523651 Ki = 0.21 nM T89034 CH0N9A 155523885 Ki = 0.32 nM T89034 CYL8M0 155526377 Ki = 5.2 nM T89034 CX7CO2 155527010 Ki = 0.13 nM T89034 CI1FR2 155529536 Ki = 0.48 nM T89034 C46AZL 155530642 Ki > 25000 nM T89034 CP8K2J 155531811 Ki = 22.7 nM T89034 C0UR8Q 155531991 Ki = 5.9 nM T89034 C8MUD0 155533285 IC50 = 660000 nM T89034 CX85KR 155535433 Ki = 1.2 nM T89034 CIHM01 155535907 Ki = 19.7 nM T89034 C0OHB7 155537066 IC50 = 140000 nM T89034 C7JMK4 155538439 Ki = 0.07 nM T89034 C9QE5N 155538514 Ki = 2.69 nM T89034 CRMS15 155539823 Ki = 1.8 nM T89034 CRT3D4 155540148 Ki = 0.77 nM T89034 CEM6G9 155540636 Ki = 8.3 nM T89034 CL90DN 155540666 Ki = 28 nM T89034 C4CHR9 155542229 Ki = 8 nM T89034 C4P2GV 155543617 Ki > 25000 nM T89034 C8Q9FS 155544416 Ki = 5000 nM T89034 CH2S6R 155546346 Ki > 10000 nM T89034 CSI5J1 155548907 Ki = 81.3 nM T89034 CU9FL4 155551858 Ki = 0.041 nM T89034 CA5VG2 155552651 Ki = 12.8 nM T89034 C5S6HO 155553129 Ki = 0.77 nM T89034 C5TV4J 155554082 Ki = 61.1 nM T89034 C9F5GQ 155555101 Ki = 2 nM T89034 CU8LR3 155555208 Ki > 25000 nM T89034 CNA52L 155557444 Ki = 16 nM T89034 CXL5D4 155558368 Ki = 0.54 nM T89034 CYTL03 155559627 Ki = 2.5 nM T89034 CNZ1K5 155559920 Ki > 10000 nM T89034 C3SXY1 155561904 Ki = 50.6 nM T89034 C14VGQ 155562325 Ki = 4.7 nM T89034 CX5O7K 155562968 Ki = 0.51 nM T89034 CWV02J 155565423 Ki = 0.45 nM T89034 CMF0N3 155565737 Ki = 16 nM T89034 CP4F1U 155567613 Ki = 0.14 nM T89034 CI08UH 155567722 Ki = 3.3 nM T89034 CEZ8B9 155568406 Ki = 4540 nM T89034 CK0EA2 155568484 Ki = 0.45 nM T89034 CS7NI8 155569220 Ki = 0.61 nM T89034 C2GES3 2037 IC50 = 7 ug.mL-1 T89034 CVK8X3 44338049 IC50 = 0.23 nM T89034 CD81GH 46830813 IC50 = 490 nM T89034 CL2S7B 90655701 Ki = 1150000 nM T89034 D00KJP 10322586 Ki = 4400 nM T89034 D00PEJ 16658631 Ki = 3200 nM T89034 D00POF 21707121 Ki = 1216 nM T89034 D01JUI 44339119 Ki = 7300 nM T89034 D01LCS 447480 Ki = 600 nM T89034 D02AVL 18376720 Ki > 5000 nM T89034 D02PAU 16731825 Ki > 10000 nM T89034 D02YIW 1794 IC50 > 10000 nM T89034 D03ZUM 6917805 IC50 = 190 nM T89034 D05SVA 125520 IC50 = 800 nM T89034 D06AVE 10200844 Ki = 1302 nM T89034 D06CJP 16658353 Ki > 100000 nM T89034 D06HOI 44249821 Ki > 16000 nM T89034 D06MTX 1506 Ki = 46000 nM T89034 D07SFI 2332 Ki = 350000 nM T89034 D07ZRG 46899577 Ki = 39 nM T89034 D08KCA 72429 IC50 = 1200 nM T89034 D08OCL 44331823 Ki > 400000 nM T89034 D09EVY 10797510 IC50 = 5700 nM T89034 D09TNA 44332077 Ki = 164000 nM T89034 D0A8WP 447732 Ki = 1950 nM T89034 D0EH1F 44332057 Ki > 100000 nM T89034 D0F2YC 10038543 IC50 = 2900 nM T89034 D0F6EZ 44436702 Ki > 1000000 nM T89034 D0J1CC 11948634 Ki > 13000 nM T89034 D0J1QT 44473100 Ki > 16000 nM T89034 D0J2SM 296008 IC50 = 6680 nM T89034 D0JU9N 6914623 Ki > 2800 nM T89034 D0K0GU 44392430 Ki = 134 nM T89034 D0K4PK 16658352 Ki = 13000 nM T89034 D0K7YL 447476 Ki = 100 nM T89034 D0M2PE 29012033 Ki = 844000 nM T89034 D0MQ6K 10574241 Ki = 4700 nM T89034 D0N1PW 134348 Ki = 111000 nM T89034 D0ON2Z 204102 Ki > 2300 nM T89034 D0R9CH 3400921 Ki > 10000 nM T89034 D0S4MQ 44392405 Ki = 1350 nM T89034 D0SP2I 6852210 Ki = 20000 nM T89034 D0Y5IQ 44255320 IC50 = 10000 nM T89034 D0Y8QU 9869156 IC50 > 2500 nM T89034 D0Y9PH 45486355 Ki = 6000 nM T89034 D0Z7YI 44331573 Ki = 61500 nM T35640 D07DJQ 10219 IC50 > 50 ug.mL-1 T35640 D0DJ4A 5311281 IC50 = 5.5 ug.mL-1 T35640 D0GT8W 11635371 IC50 = 18 nM T35640 CIDV34 180535 IC50 > 50000 nM T35640 CQOE70 442195 IC50 > 10 ug.mL-1 T35640 CU09IZ 5281318 IC50 = 1360 nM T35640 CTLO76 5281321 IC50 = 950 nM T35640 CTQD52 9805155 IC50 = 105 nM T35640 C27AQC 9912035 IC50 = 40 nM T35640 CYKV73 9934394 IC50 = 140 nM T35640 C6H4MG 10324921 IC50 = 1.4 nM T35640 CZR76O 10437814 IC50 = 3 nM T35640 CH2M7K 10482211 IC50 = 5 nM T35640 C01OXC 10863710 IC50 = 295 nM T35640 CJ86FE 10907156 IC50 = 7 nM T35640 CEKM83 10940028 IC50 = 6 nM T35640 C5VCE2 10940362 IC50 > 20000 nM T35640 C8RCW6 10950607 IC50 = 145 nM T35640 C8FB9V 10950903 IC50 = 10 nM T35640 CMF19U 10951666 IC50 = 3750 nM T35640 CE25DA 10960604 IC50 > 20000 nM T35640 CK21DB 10961634 IC50 = 8 nM T35640 C6Y2DN 10962022 IC50 = 55 nM T35640 C57QXY 11006190 IC50 = 5 nM T35640 CH13VS 11026262 IC50 = 10 nM T35640 CD9G5Y 11026412 IC50 = 1400 nM T35640 C5BO3A 11026764 IC50 = 30 nM T35640 CSJ28E 11038325 IC50 = 7 nM T35640 CBC9Q4 11049285 IC50 = 50 nM T35640 C0YXT9 11058089 IC50 = 90 nM T35640 C8GJ5Z 11059518 IC50 > 20000 nM T35640 C7Z4ET 11059680 IC50 > 20000 nM T35640 CU25JB 11070521 IC50 = 8 nM T35640 CA7Z0K 11080780 IC50 > 20000 nM T35640 C4HC9O 11090982 IC50 = 3900 nM T35640 CQD40Z 11092636 IC50 = 5 nM T35640 CU6G1R 11133700 IC50 = 10700 nM T35640 C9E7UF 11134408 IC50 = 265 nM T35640 C2TN7V 11143616 IC50 = 150 nM T35640 C2RVI8 11144584 IC50 = 4300 nM T35640 CY9ZS1 11145114 IC50 = 139 nM T35640 C1KY6C 11399131 IC50 = 260 nM T35640 C5ECV1 11699447 IC50 = 2.5 nM T35640 CG2X8S 11755267 IC50 = 6 nM T35640 CMCY42 11784188 IC50 = 9100 nM T35640 CT6JM8 11964801 IC50 = 650 nM T35640 C5U3GA 15944763 IC50 = 300 nM T35640 CS09UY 44358322 IC50 = 115 nM T35640 CNP8V6 44465635 IC50 = 69 nM T35640 C0RET8 44465882 IC50 = 550 nM T35640 C50AQV 46220742 IC50 = 11 nM T35640 C7PQ3D 46220743 IC50 = 1260 nM T35640 C8KW5U 46220745 IC50 = 13 nM T35640 CWT86L 46220746 IC50 = 50 nM T35640 CZ45LI 46220747 IC50 = 56 nM T35640 CN82EM 46220960 IC50 = 26 nM T35640 C5XW8J 46220961 IC50 = 8 nM T35640 CW7GT5 46220962 IC50 = 12 nM T35640 C3EQD6 46220963 IC50 = 240 nM T35640 CLB08M 46220964 IC50 = 170 nM T35640 C84NLX 46221188 IC50 = 58 nM T35640 C8RLT6 46221189 IC50 = 4.8 nM T35640 CQCX63 46221190 IC50 = 6 nM T35640 CBJ9D8 46221191 IC50 = 400 nM T35640 CHR8C9 46221192 IC50 = 80 nM T35640 CX69AF 46221417 IC50 = 4.4 nM T35640 CL6W2J 46224084 IC50 = 11 nM T35640 C1PV5C 46224085 IC50 = 80 nM T35640 CPL12F 46224086 IC50 = 60 nM T35640 C82LCY 46224087 IC50 = 12 nM T35640 CLB5Y2 46224088 IC50 = 80 nM T35640 CLP8U2 49864499 IC50 = 1200 nM T35640 C4KO3T 49864502 IC50 = 1600 nM T35640 CB4LK6 49864524 IC50 = 240 nM T35640 CWL20A 49864525 IC50 = 430 nM T35640 CS1P8W 49864598 IC50 = 3800 nM T35640 C7P8CR 90645221 IC50 > 10000 nM T35640 C9NGQ3 90645222 IC50 = 7900 nM T35640 CW0IE7 90645223 IC50 = 488 nM T35640 COAL72 90645224 IC50 > 10000 nM T35640 CR54SJ 90645225 IC50 = 37 nM T35640 CH96PL 90645226 IC50 = 358 nM T35640 C5EQX8 90645227 IC50 > 10000 nM T35640 CXZ34D 90645228 IC50 = 65 nM T35640 C1B9AV 90645229 IC50 = 100 nM T35640 C3UO8P 90645230 IC50 = 28 nM T35640 CTZ27J 90645231 IC50 = 16 nM T35640 C35WKV 90645232 IC50 = 117 nM T35640 C5JNP3 90645233 IC50 = 23 nM T35640 CYLC62 90645234 IC50 = 22 nM T35640 CGE38T 90645235 IC50 = 12900 nM T35640 CRS82Y 90645236 IC50 = 180 nM T35640 D07XCA 9846729 IC50 = 44 nM T37847 D0OT0O 44561 IC50 = 74000 nM T37847 D05RQB 457964 IC50 = 500 nM T37847 CQ87XE 72187 IC50 = 3300 nM T37847 C1NZG5 73183 IC50 > 500000 nM T37847 CO6HK2 73185 IC50 > 500000 nM T37847 CU3P0Y 484047 IC50 = 300 nM T37847 C61SXL 492406 IC50 = 600 nM T37847 CZ1A8T 503580 IC50 = 1200 nM T37847 CU1JO9 512102 IC50 = 97000 nM T37847 C41FNP 512104 IC50 = 39000 nM T37847 CAB9E5 512105 IC50 = 44000 nM T37847 CAWB10 512106 IC50 > 500000 nM T37847 C3N5TL 512107 IC50 > 500000 nM T37847 CD6X0S 512108 IC50 > 500000 nM T37847 C70CDA 512109 IC50 > 500000 nM T37847 CFTL84 512110 IC50 > 500000 nM T37847 C64WVM 512111 IC50 > 500000 nM T37847 C9Z5QH 512112 IC50 > 500000 nM T37847 CBX73L 512113 IC50 > 500000 nM T37847 C4I3CT 512114 IC50 > 500000 nM T37847 C7BJ0D 512115 IC50 > 500000 nM T37847 CQ1M8B 512116 IC50 > 500000 nM T37847 C4OHD3 512117 IC50 > 500000 nM T37847 CI2VD7 512118 IC50 > 500000 nM T37847 CVO12S 512121 IC50 > 500000 nM T37847 C3XUT4 512122 IC50 > 500000 nM T37847 CK52PA 512123 IC50 > 500000 nM T37847 CJV43L 512124 IC50 > 500000 nM T37847 CC7FO5 512125 IC50 > 500000 nM T37847 CKJ47G 512126 IC50 > 500000 nM T37847 C8F1DN 6482394 IC50 = 500 nM T37847 COS5K6 13077901 IC50 > 500000 nM T37847 CJ4S7I 13077902 IC50 > 500000 nM T37847 CW2C3A 13077914 IC50 > 500000 nM T37847 CFVJ31 13077915 IC50 > 500000 nM T37847 CK8SV1 13077916 IC50 = 79000 nM T37847 C9F4DN 13077917 IC50 = 87000 nM T37847 C0H1VN 13077918 IC50 = 90000 nM T37847 CHQ54B 13077919 IC50 > 500000 nM T37847 CPT13F 13077920 IC50 = 73000 nM T37847 CY0XB6 13077921 IC50 > 500000 nM T37847 CA3L0J 13077922 IC50 > 500000 nM T37847 C9WER8 13077924 IC50 > 500000 nM T37847 CMLY18 13077925 IC50 > 500000 nM T37847 CH0V3D 13077926 IC50 > 500000 nM T37847 C3QXW6 13077927 IC50 > 500000 nM T37847 CRK6T2 13077928 IC50 > 500000 nM T37847 CI1C0H 13077929 IC50 > 500000 nM T37847 CSL6Z2 13077930 IC50 = 250000 nM T37847 C3XC0A 13077932 IC50 > 500000 nM T37847 CV6Q3M 23679405 IC50 > 500000 nM T37847 CX76DA 23679406 IC50 > 500000 nM T37847 CV06UD 23679407 IC50 > 500000 nM T37847 CH2RO0 23679408 IC50 > 500000 nM T37847 C8OZ4G 23679409 IC50 > 500000 nM T37847 CN2J1S 23679410 IC50 > 500000 nM T37847 CT0PX1 23679411 IC50 = 165000 nM T37847 CGC0V3 23679412 IC50 > 500000 nM T37847 CIS13H 23679413 IC50 = 500000 nM T37847 C5VXS7 23679414 IC50 = 52000 nM T37847 CDXU03 23679415 IC50 = 54000 nM T13075 D09XZB 123631 IC50 > 50000 nM T13075 D0E6XR 3062316 IC50 < 1 nM T13075 D0R0MW 5329102 IC50 < 1 nM T13075 D0W5HK 216239 IC50 = 250 nM T13075 D05ADP 160355 IC50 = 4000 nM T13075 D07EHV 44814409 IC50 > 10000 nM T13075 D0E3TC 44259 IC50 = 3850 nM T13075 D0FD6D 11751922 IC50 = 48 nM T13075 D02VBF 25023738 IC50 = 450 nM T13075 D0T3ME 156422 IC50 > 30000 nM T13075 C8Z1FA 1960 Ki = 80000 nM T13075 CEC30Q 3674 IC50 = 1240 nM T13075 CN64JR 8323 IC50 = 4000 nM T13075 CTLV26 129236 IC50 = 10000 nM T13075 CN6AY0 491467 IC50 > 10000 nM T13075 CPQV76 5353678 IC50 = 11000 nM T13075 CLN2G8 6475560 IC50 > 10000 nM T13075 CXBU49 11502255 IC50 = 1100 nM T13075 CACS26 11561968 Ki > 2000 nM T13075 CJ9KN7 11683817 IC50 > 10000 nM T13075 CU0E8O 11690457 Ki > 2000 nM T13075 CB0AP2 11705863 Ki > 2000 nM T13075 C3YRU7 15295578 IC50 = 250 nM T13075 C5VPH9 16129448 IC50 = 872 nM T13075 CL81VC 21100709 IC50 = 78800 nM T13075 C7YG1N 24759534 IC50 = 230 nM T13075 CHU23B 25168304 IC50 = 14 nM T13075 C3VRO9 44557921 IC50 = 9120.11 nM T13075 CF90OX 44576212 IC50 = 1300 nM T13075 CLS29B 46872626 IC50 > 10000 nM T13075 C29PHE 46882055 IC50 = 14 nM T13075 CRLZ94 46912952 IC50 = 600 nM T13075 C1VA0B 46912953 IC50 = 180 nM T13075 C1PG7E 46912955 IC50 = 150 nM T13075 CBS64G 49830252 IC50 = 12000 nM T13075 CD2K4R 50908681 Ki > 1000000 nM T13075 CM42BY 51000510 Ki > 1000000 nM T13075 C8NA4L 53384644 IC50 > 30000 nM T13075 C4S1HX 56589672 IC50 = 1500 nM T13075 CON8H1 59326984 IC50 = 12100 nM T13075 CXJ63M 59603829 IC50 = 630 nM T13075 CQEU96 59603842 IC50 = 2100 nM T13075 C1MR8Q 60097495 IC50 > 10000 nM T13075 CIM7H1 66575095 IC50 = 251 nM T13075 C37NKO 67129970 IC50 = 5220 nM T13075 CK80LJ 67130050 IC50 = 7540 nM T13075 CV63UL 67240318 IC50 > 10000 nM T13075 C7GRV2 68755406 IC50 > 10000 nM T13075 C5DGR9 69036886 IC50 = 10000 nM T13075 C8CK9I 70682868 IC50 = 78 nM T13075 C3WK5U 70684923 IC50 = 660 nM T13075 CZQX81 70684935 IC50 > 10000 nM T13075 C2MPQ3 70686838 IC50 = 7580 nM T13075 C7B0ZJ 70687101 IC50 > 10000 nM T13075 C1MCQ3 70691009 IC50 = 8820 nM T13075 CCJH52 70691010 IC50 = 5490 nM T13075 CHN63I 70691266 IC50 = 2470 nM T13075 CAJF37 70693140 IC50 = 4670 nM T13075 C2U7ES 70693141 IC50 = 19700 nM T13075 CQ75AH 70693142 IC50 = 9180 nM T13075 C5S8ZN 70693380 IC50 = 142 nM T13075 CC48LS 70695212 IC50 = 3540 nM T13075 CN8T9F 70695463 IC50 = 390 nM T13075 C7VA0I 71450358 IC50 = 736 nM T13075 CZ2OE6 71452173 IC50 = 9 nM T13075 CSPN93 71452174 IC50 = 33 nM T13075 CR53ZS 71452175 IC50 = 174 nM T13075 CM14JZ 71452176 IC50 = 383 nM T13075 CX1KZ0 71453985 IC50 = 568 nM T13075 CFGP02 71455731 IC50 = 95 nM T13075 CS27GC 71457514 IC50 = 54 nM T13075 C16OVY 71457515 IC50 = 18500 nM T13075 C3KIM9 71461149 IC50 = 19 nM T13075 CW6MK4 71462888 IC50 = 146 nM T13075 C9V6KY 71462889 IC50 = 225 nM T13075 C0DL3F 72698602 IC50 = 469800 nM T13075 C1HW4B 89735655 IC50 = 18000 nM T13075 C2AN7T 134611886 IC50 > 100000 nM T13075 CI1E8V 137634241 IC50 > 10000 nM T13075 CS61AX 137659496 IC50 > 100000 nM T13075 C3W4RO 138403252 IC50 = 1800 nM T13075 C07EKN 138454794 IC50 > 10000 nM T13075 D00ERW 44444843 Ki > 6916 nM T13075 D00JGL 6419753 IC50 = 300 nM T13075 D01MNK 25125014 IC50 = 1040 nM T13075 D06HVH 54613583 IC50 = 330 nM T13075 D09FFE 449241 Ki = 38300 nM T13075 D0H4VB 71461150 IC50 = 442 nM T13075 D0L4WN 31420 IC50 = 4000 nM T13075 D0N3LC 90643548 IC50 = 545 nM T13075 D0RJ8J 76072859 IC50 = 694 nM T13075 D0Y6OK 6688 IC50 > 40000 nM T23666 D04TNT 46851313 EC50 > 10000 nM T23666 C61DRT 568 EC50 = 1000000 nM T23666 CT53FM 1674 EC50 = 490 nM T23666 CEB26G 2336 EC50 = 5 nM T23666 C4DS3F 2361 EC50 = 8.4 nM T23666 CG3YN1 10215 EC50 = 1700 nM T23666 CR6Z2V 15625 EC50 = 10 nM T23666 CIH70E 17097 EC50 = 130016.96 nM T23666 C9DV0T 18636 EC50 = 10000 nM T23666 C80NPE 21510 EC50 = 257039.58 nM T23666 CRS5X0 32781 EC50 = 279898.13 nM T23666 CXY3J5 35454 EC50 = 1300.17 nM T23666 CM9A7B 35823 EC50 = 9099.13 nM T23666 C86CSG 36187 EC50 = 709.58 nM T23666 CCH80P 36188 EC50 = 4265.8 nM T23666 C84TFS 36401 EC50 = 139958.73 nM T23666 CMW62N 36614 EC50 = 70.96 nM T23666 CZ3X5U 36934 EC50 = 159.96 nM T23666 CK58GW 37034 EC50 = 79432.82 nM T23666 CW6OE1 37207 EC50 = 100000 nM T23666 CZPY97 38019 EC50 = 7095.78 nM T23666 C3PB8W 38193 EC50 = 3198.9 nM T23666 CGLR53 38213 EC50 = 15.49 nM T23666 COL9W1 38251 EC50 = 279.9 nM T23666 C7CNW2 38253 EC50 = 13001.7 nM T23666 CB1IN7 38254 EC50 = 6456.54 nM T23666 CH9T6S 38439 EC50 = 79.43 nM T23666 CRVK01 39728 EC50 = 1.479 nM T23666 C4B9SE 39729 EC50 = 1.5 nM T23666 C43IJH 39732 EC50 = 794.33 nM T23666 CB7I1U 39929 EC50 = 41.02 nM T23666 CA7S5E 40479 EC50 = 15995.58 nM T23666 COU45D 42128 EC50 = 15.14 nM T23666 CDP65S 42129 EC50 = 1000 nM T23666 C53EUI 42131 EC50 = 19010.78 nM T23666 C3SC0Q 42134 EC50 = 219.79 nM T23666 C52CQR 42138 EC50 = 74.13 nM T23666 CM2LV8 42140 EC50 = 269.77 nM T23666 CPJF68 42836 EC50 = 1099.01 nM T23666 C5F0JI 42839 EC50 = 1300.17 nM T23666 C5HGM6 42840 EC50 = 199.99 nM T23666 C5H3UV 43255 EC50 = 246036.76 nM T23666 CSN94L 43495 EC50 = 46.77 nM T23666 CS15IR 44101 EC50 = 349.95 nM T23666 C0U6KL 47299 EC50 = 4720.63 nM T23666 CM39CR 47300 EC50 = 10000 nM T23666 C40ANZ 47650 EC50 = 14125.38 nM T23666 COJP23 49923 EC50 = 119.95 nM T23666 CD0H7K 49931 EC50 = 8298.51 nM T23666 C07RVD 50610 EC50 = 3097.42 nM T23666 CB5DR9 50891 EC50 = 5000.35 nM T23666 CI0HV2 51043 EC50 = 27989.81 nM T23666 CA76OQ 51126 EC50 = 199.99 nM T23666 CG5B9U 51130 EC50 = 230.14 nM T23666 CSV54H 51464 EC50 = 19998.62 nM T23666 CE6P9Q 53036 EC50 = 4102.04 nM T23666 CL8Q9G 53154 EC50 = 1000000 nM T23666 C61WDC 53524 EC50 = 85113.8 nM T23666 C3F5RQ 55103 EC50 = 349.95 nM T23666 CV68SN 55104 EC50 = 219.28 nM T23666 CPGM67 55111 EC50 = 25.12 nM T23666 CS43GX 55112 EC50 = 199.99 nM T23666 C1Z8QO 55119 EC50 = 4365.16 nM T23666 C15UKH 55125 EC50 = 449.78 nM T23666 CA2E4M 55130 EC50 = 67.76 nM T23666 C46SXT 55133 EC50 = 399.94 nM T23666 CSX23L 60059 EC50 = 295.12 nM T23666 C7D9CG 60312 EC50 = 6.607 nM T23666 CYIT27 63078 EC50 = 99083.19 nM T23666 CY5KZ7 63090 EC50 = 130.02 nM T23666 C9E4UL 86291 EC50 = 92.9 nM T23666 C1A7HF 108120 EC50 = 1.169 nM T23666 CZG7F5 114896 EC50 = 11.51 nM T23666 CQOJ45 114900 EC50 = 49 nM T23666 CY38KF 115206 EC50 = 219.79 nM T23666 CC62AF 161166 Ki = 21600 nM T23666 CGS23D 176111 EC50 = 0.4467 nM T23666 CHQU87 184065 EC50 = 2 nM T23666 C6FB9I 184066 EC50 = 16.98 nM T23666 CLSO47 527713 EC50 = 41975.9 nM T23666 CWAM07 688681 EC50 = 270 nM T23666 CFO1Z7 1778614 IC50 = 2.6 nM T23666 CP69KZ 5324349 EC50 = 1340 nM T23666 CX23PO 6020016 IC50 = 7600 nM T23666 CHE70V 9838722 Ki = 831763771.1 nM T23666 CUCM03 10062125 Ki = 714496326.1 nM T23666 C2V4ZO 10265357 EC50 = 270 nM T23666 C40NPC 10407651 Ki = 476430986.8 nM T23666 CB9JS4 10565123 EC50 > 10000 nM T23666 C6DJQ9 10900930 EC50 = 215 nM T23666 CIG8Z6 11153316 Ki = 16672472.13 nM T23666 C9T6KS 11197891 Ki = 52722986.14 nM T23666 CO2N4Z 11208222 Ki = 175388050.2 nM T23666 CN6V7O 11209303 Ki = 147231250.2 nM T23666 C7M9AJ 11230651 Ki = 10423174.29 nM T23666 CQHW46 11243890 Ki = 12 nM T23666 C3B4HX 11244016 Ki = 71449632.61 nM T23666 CZ1LG3 11266077 Ki = 12 nM T23666 C8LFT9 11287739 Ki = 263633138.6 nM T23666 CY2GB4 11300595 Ki = 199986187 nM T23666 CP61NH 11310856 Ki = 15885467.49 nM T23666 CW3L1T 11358876 Ki = 50118723.36 nM T23666 CL8JI2 11391816 Ki = 41686938.35 nM T23666 C0L2IW 11414230 Ki = 322849412.2 nM T23666 CYM9V2 11414783 Ki = 12 nM T23666 C9YW0P 11425113 Ki = 108893009.3 nM T23666 CYIU98 11438491 Ki = 200447202.7 nM T23666 CP4M8J 11482995 Ki = 12 nM T23666 CS4X7T 11817441 Ki = 45498806.02 nM T23666 CU6D9M 12989853 EC50 = 94 nM T23666 CZXD09 46232106 EC50 > 10000 nM T23666 CW19MT 46232107 EC50 = 330 nM T23666 CR1SN4 46232174 EC50 = 200 nM T23666 C1JVS0 46232175 EC50 = 450 nM T23666 CJ3FM4 46925833 EC50 = 7300 nM T23666 C87GEW 102435977 IC50 = 1500 nM T23666 C14SPM 118709590 EC50 = 93 nM T23666 CG87VT 118709591 EC50 = 320 nM T23666 C7UT4N 118709592 EC50 = 230 nM T23666 CJP13G 118709593 EC50 = 55 nM T23666 CV0ES8 118709594 EC50 > 6700 nM T23666 CD3MA2 118709595 EC50 = 86 nM T23666 CI3X9L 127049803 EC50 = 630 nM T23666 C2O5LX 127049804 EC50 = 2300 nM T23666 CEVL69 135423792 IC50 = 20000 nM T23666 C7RH0P 135423823 IC50 = 5200 nM T23666 CB2WH3 135423824 IC50 = 25000 nM T23666 CQKV19 135423826 IC50 > 30000 nM T23666 CO7DF9 135423833 IC50 = 5400 nM T23666 CR9JW4 135423834 IC50 > 30000 nM T23666 C98KOZ 135423836 IC50 = 18800 nM T23666 C1V8BA 135423843 IC50 = 13000 nM T23666 C6W3IR 135423846 IC50 = 24000 nM T23666 CUT84A 155568798 EC50 > 50000 nM T23666 D01SHB 3845 EC50 = 300 nM T23666 D03NTD 9878556 Ki = 12 nM T23666 D0B3ZB 135398521 EC50 = 160 nM T23666 D0G3TK 5280863 IC50 = 28 nM T23666 D0O9NE 5388063 Ki = 130016957.8 nM T77236 D0V3YT 10324367 IC50 = 1100 nM T77236 D0X9CH 3010818 IC50 > 10000 nM T77236 D0J6AU 10152654 IC50 = 795 nM T77236 C0XQP7 6917747 IC50 > 100000 nM T77236 CN26IL 9547980 Ki > 30000 nM T77236 CILB73 11649751 Ki > 20000 nM T77236 C31MCN 13186896 IC50 > 100000 nM T77236 C9LW6H 15985754 IC50 = 0.3 nM T77236 C6XPN4 16664855 IC50 = 331 nM T77236 CQU38W 24900755 IC50 = 5908 nM T77236 C2S8VB 24901099 IC50 = 487 nM T77236 CIN28B 24901100 IC50 = 3760 nM T77236 CD2EH0 24901101 IC50 = 1826 nM T77236 CS7B3F 24901102 IC50 > 10000 nM T77236 CL96WQ 42633150 IC50 = 147 nM T77236 CZ5F4C 42633340 IC50 = 76 nM T77236 C5XV0H 42633341 IC50 = 4 nM T77236 CZS24P 42633520 IC50 = 16 nM T77236 CI78XT 42633521 IC50 = 56 nM T77236 CU6PL7 42633691 IC50 = 64 nM T77236 CQ9TR8 42633692 IC50 = 67 nM T77236 C6FJW2 42634249 IC50 = 22 nM T77236 C9EN0G 42634411 IC50 = 37 nM T77236 C2ZXJ7 42634578 IC50 = 174 nM T77236 CI25RJ 42634754 IC50 = 51 nM T77236 CZ6B1F 42635119 IC50 = 23 nM T77236 C5X4WG 42635483 IC50 = 12 nM T77236 CZ56BP 44263398 IC50 > 20000 nM T77236 CS6X7V 44426055 IC50 > 10000 nM T77236 C8IB2W 44426056 IC50 > 100000 nM T77236 C4YAJ7 46228924 IC50 > 10000 nM T77236 C4I0JY 50925524 IC50 = 4 nM T77236 C7DO0F 52941283 IC50 = 80 nM T77236 CU1TW6 52941414 IC50 = 769 nM T77236 C9MK7J 52942931 IC50 = 547 nM T77236 C4TY6S 52943722 IC50 > 10000 nM T77236 CQ6N0I 52943841 IC50 > 10000 nM T77236 CV8L9Z 52945985 IC50 = 24 nM T77236 CLJ83U 52946267 IC50 = 3242 nM T77236 CT28XU 52947761 IC50 = 654 nM T77236 CLX2Y4 60148518 Ki > 40000 nM T77236 C0DA6M 60166364 Ki > 40000 nM T77236 C4G1SF 60166365 Ki > 40000 nM T77236 COM7U3 60166366 Ki > 4000 nM T77236 COQ82A 60166367 Ki > 4000 nM T77236 C2Y7EK 60166492 Ki > 4000 nM T77236 C4PHR1 60166493 Ki > 4000 nM T77236 CG4DZ7 60166494 Ki > 4000 nM T77236 C5E2PB 60166495 Ki = 3200 nM T77236 CXD39V 60166496 Ki > 4000 nM T77236 CM8XO5 60166497 Ki > 4000 nM T77236 D06WQP 60148519 Ki = 21 nM T18474 D0E3TC 44259 IC50 = 21.5 nM T18474 D0T3ME 156422 IC50 = 90 nM T18474 C8NA4L 53384644 IC50 > 30000 nM T18474 CV63UL 67240318 IC50 > 10000 nM T18474 C0Y8ZK 91933875 IC50 > 1000 nM T18474 C9WGB8 127035904 IC50 = 2600 nM T18474 C2MD1Q 155513187 IC50 > 10000 nM T18474 D05FXD 44478401 IC50 = 3 nM T18474 D0X8BU 71718651 IC50 = 2400 nM T44861 D0AZ3C 5291 IC50 > 100000 nM T44861 D0E6XR 3062316 IC50 > 50000 nM T44861 D0E9KA 6918670 EC50 = 4.1 nM T44861 D09DHT 27924 Ki = 0.8 nM T44861 D0E3TC 44259 IC50 = 5.5 nM T44861 D0E6AH 5280757 Ki = 0.44 nM T44861 D0I6VU 176167 IC50 = 1000 nM T44861 D0LF1U 5287969 IC50 = 890 nM T44861 D0MS3Z 16725726 IC50 = 14 nM T44861 D0W3LI 153999 IC50 = 250 nM T44861 D03BNU 59604787 IC50 > 10000 nM T44861 D0LF0O 135441202 IC50 = 20300 nM T44861 D0R1JI 5281847 IC50 = 3000 nM T44861 D0WS1V 448991 IC50 > 100000 nM T44861 D01EFO 9864718 IC50 > 500000 nM T44861 D0R2TM 5287736 IC50 = 20 nM T44861 D0T3ME 156422 IC50 = 1900 nM T44861 C8OI7N 2290 IC50 = 16 nM T44861 CJ17AM 4877 IC50 > 100000 nM T44861 C2EWT0 72425 Ki = 0.32 nM T44861 CG2P1X 159320 Ki = 0.8 nM T44861 C8PU1O 188534 Ki = 0.46 nM T44861 CMN15U 192686 IC50 = 42000 nM T44861 CT09IC 455726 Ki = 1.8 nM T44861 C0G6JH 455733 Ki = 410 nM T44861 C6DLK3 644364 IC50 = 2600 nM T44861 CTID76 5282335 IC50 = 45000 nM T44861 CLA43B 5327919 IC50 = 90 nM T44861 CPDC54 5327920 IC50 = 50 nM T44861 CCB9G3 5327921 IC50 = 5 nM T44861 CRTQ98 5327922 IC50 = 0.9 nM T44861 CP20NQ 5327923 IC50 = 20 nM T44861 C98CNM 5327943 IC50 = 410 nM T44861 C61URB 5327944 IC50 = 0.9 nM T44861 CWUY53 5327945 IC50 = 4200 nM T44861 CQ54BE 5327946 IC50 = 40 nM T44861 CIB3P0 5327947 IC50 = 30 nM T44861 CVG0A1 5327948 IC50 = 3 nM T44861 C8M3PD 5327949 IC50 = 410 nM T44861 CA25BM 5327950 IC50 = 22000 nM T44861 COP0Q2 5327951 IC50 = 270 nM T44861 CB47VN 5327952 IC50 = 130 nM T44861 CPO51K 5327953 IC50 = 30 nM T44861 CI6AY9 5327954 IC50 = 820 nM T44861 C1Q0PM 5327955 IC50 = 1900 nM T44861 CXA23M 5327956 IC50 = 220 nM T44861 CH73DT 5327957 IC50 = 290 nM T44861 CTI6K8 5327963 IC50 = 300 nM T44861 CAO1N9 5327979 IC50 = 20 nM T44861 CMP3X8 5327994 IC50 < 50 nM T44861 C4DG8Y 5327995 IC50 = 30 nM T44861 CDL0S2 5327996 IC50 = 4400 nM T44861 CC43JH 5327997 IC50 = 420 nM T44861 CKS8M6 5327998 IC50 = 20 nM T44861 CQ7OZ6 5327999 IC50 = 90 nM T44861 CQWO93 5328000 IC50 = 130 nM T44861 CU73IX 5328002 IC50 = 18 nM T44861 CTVP40 5328003 IC50 = 50 nM T44861 CBSP34 5328004 IC50 = 80 nM T44861 CS78OD 5328005 IC50 = 200 nM T44861 CO9YQ6 5328006 IC50 = 310 nM T44861 CVX2L3 5328007 IC50 = 10 nM T44861 CPD1U9 5328008 IC50 = 24 nM T44861 C3X6QJ 5328012 IC50 = 67 nM T44861 CZO4E1 5328013 IC50 = 50 nM T44861 C2RA4O 5352033 Ki = 0.2 nM T44861 CF32UV 5471818 Ki = 1.16 nM T44861 CW1ZY2 6520576 Ki = 0.9 nM T44861 CG17TN 6914611 IC50 = 6100 nM T44861 C7E2QK 6914613 IC50 = 930 nM T44861 C0IK9O 9543716 EC50 = 7490 nM T44861 CZR3M4 9799152 IC50 > 100000 nM T44861 C4PA5X 9800852 Ki = 1630 nM T44861 CI3O6X 9814609 IC50 > 500000 nM T44861 CX9DG5 9822042 IC50 > 500000 nM T44861 C8J1OL 9826373 IC50 = 400 nM T44861 CSH0A9 9847014 IC50 = 4400 nM T44861 C3UQL7 9860872 IC50 > 500000 nM T44861 CCJK12 9865633 Ki = 10.7 nM T44861 C20NKA 9889351 IC50 = 400 nM T44861 C2TC1L 9910609 IC50 > 125000 nM T44861 CUKH27 9943194 IC50 > 500000 nM T44861 CU78NO 9947433 IC50 = 17000 nM T44861 CP5NJ3 9952970 Ki = 14.6 nM T44861 CYT7R9 9953676 IC50 > 100000 nM T44861 CV34AB 9958125 IC50 = 6000 nM T44861 CJ40GO 9965429 IC50 > 500000 nM T44861 C2W3AV 9995236 IC50 = 1200 nM T44861 CY65CO 10030073 IC50 = 5 nM T44861 C2UGV9 10030483 IC50 = 90 nM T44861 C0G5DK 10039959 IC50 > 100000 nM T44861 C7YD1X 10048045 IC50 > 25000 nM T44861 CS2ZL3 10090448 Ki = 290 nM T44861 CG7JO8 10099482 IC50 = 90 nM T44861 C93LPQ 10099652 IC50 = 110 nM T44861 C63CFD 10111108 IC50 > 500000 nM T44861 CL42XS 10136330 IC50 > 500000 nM T44861 C2O7ZH 10137972 IC50 = 1.8 nM T44861 C76TVG 10143584 IC50 = 2200 nM T44861 CUW34X 10157645 IC50 > 500000 nM T44861 C7JP1A 10163439 IC50 = 250 nM T44861 COC30E 10181160 IC50 > 500000 nM T44861 CJN72C 10185160 IC50 = 86 nM T44861 CJ0R2G 10187378 IC50 = 1500 nM T44861 CGOT91 10207821 IC50 = 350 nM T44861 C51SKM 10209082 IC50 = 490 nM T44861 C8W2HS 10224497 Ki = 91.1 nM T44861 C3VK7T 10229967 IC50 = 1160 nM T44861 C7SFI1 10296883 IC50 = 1.3 nM T44861 CAX9W2 10302405 IC50 = 31 nM T44861 CFW0U4 10316976 Ki = 6500 nM T44861 CFU05J 10339055 Ki = 12000 nM T44861 CFU38G 10363814 Ki = 415 nM T44861 CEH41V 10392789 IC50 = 6 nM T44861 C3RBY8 10395226 Ki = 2.5 nM T44861 CDR7X8 10415328 IC50 = 49000 nM T44861 CQXJ51 10425978 Ki = 67.5 nM T44861 CB2H1W 10451697 Ki = 2700 nM T44861 C36QRS 10453829 Ki = 92 nM T44861 C10PAC 10460251 IC50 = 4 nM T44861 C25LDK 10460643 IC50 = 32000 nM T44861 C1VI3E 10477747 IC50 = 183 nM T44861 CMA4J8 10479260 Ki = 150 nM T44861 CX7S8N 10482293 IC50 = 5 nM T44861 C78FPR 10501266 IC50 = 1400 nM T44861 C76QGP 10506540 IC50 = 6 nM T44861 CSR8Y5 10527068 IC50 = 2600 nM T44861 CDNP37 10530708 IC50 = 20 nM T44861 C5EYJ3 10554684 IC50 = 420 nM T44861 C71UIS 10555532 IC50 = 4000 nM T44861 CC0NY5 10619307 Ki = 5100 nM T44861 CI5W2K 10620066 Ki = 19 nM T44861 CZ8UA9 10650891 IC50 = 880 nM T44861 C69QNR 10665157 Ki = 1700 nM T44861 C7BTD6 10666255 Ki = 0.8 nM T44861 CJOU71 10671412 IC50 = 170 nM T44861 CM5B6A 10673286 IC50 = 2000 nM T44861 CAVX96 10686149 IC50 > 500000 nM T44861 CU6G5Y 10708835 IC50 > 500000 nM T44861 CN9I6T 10768377 IC50 = 2800 nM T44861 CL8VH3 10768554 IC50 = 7800 nM T44861 C5YMK8 10769011 IC50 = 20 nM T44861 C2TJ9X 10807429 Ki = 65 nM T44861 C7HPA0 10864309 IC50 = 7000 nM T44861 C1DRE5 10884145 IC50 = 23 ug.mL-1 T44861 C2G5CU 10894726 Ki = 1155 nM T44861 C1L4ZC 10940039 IC50 = 4200 nM T44861 CR47CD 11025838 Ki = 149 nM T44861 C67CSJ 11201611 IC50 = 17 nM T44861 CH7D3X 11233762 IC50 = 19000 nM T44861 C3ROM0 11247414 IC50 = 303 nM T44861 CBOP58 11293798 Ki > 10000 nM T44861 CANY24 11311217 IC50 = 39000 nM T44861 CRZ38O 11315034 IC50 = 92 nM T44861 CS46BW 11361072 Ki = 1457 nM T44861 C4ON7Z 11362429 IC50 = 9.4 nM T44861 C26BZX 11362471 Ki > 10000 nM T44861 C3OCV2 11371778 IC50 = 34000 nM T44861 CWXB93 11397177 Ki > 10000 nM T44861 CWM18I 11406175 IC50 > 50000 nM T44861 C1WXC5 11417488 IC50 = 50000 nM T44861 C3EXM4 11440028 IC50 = 23000 nM T44861 C64IGY 11448608 Ki > 5000 nM T44861 C8DNQ2 11453012 IC50 = 400 nM T44861 CJC95A 11454205 IC50 > 10000 nM T44861 C7I6AG 11474111 IC50 = 24000 nM T44861 C4YO9P 11516650 Ki = 1.4 nM T44861 C3KAC4 11538477 IC50 > 316 nM T44861 CTG83F 11539329 Ki > 8900 nM T44861 C1CD2N 11547825 IC50 = 292 nM T44861 C9OV5S 11561609 IC50 = 79 nM T44861 CZJY10 11574218 Ki = 2140 nM T44861 CD7PF5 11574473 IC50 > 316 nM T44861 CMIL86 11590363 Ki > 8900 nM T44861 CA9XJ2 11604381 IC50 = 15 nM T44861 CI9HQ2 11624816 IC50 > 316 nM T44861 C2LQI8 11624847 Ki = 1890 nM T44861 CK34LS 11632737 IC50 > 40000 nM T44861 CG60NH 11638724 IC50 = 33200 nM T44861 CQ5S3G 11639520 IC50 > 316 nM T44861 C9T6SC 11640926 Ki > 8900 nM T44861 CV2KF5 11646797 Ki = 980 nM T44861 C7VLD4 11654176 Ki = 3.13 nM T44861 C0WHV8 11696960 Ki = 20.6 nM T44861 CFJ4I7 11723151 IC50 = 21000 nM T44861 CCX53Q 11729563 IC50 = 400 nM T44861 C7C2FM 11737638 IC50 = 23000 nM T44861 CN0DO9 11749385 Ki = 3473 nM T44861 C47VYQ 11795964 Ki = 14 nM T44861 CM10YB 11799388 IC50 = 3300 nM T44861 CTN96I 11851810 IC50 = 0.4 nM T44861 CA05OS 11972484 IC50 = 340 nM T44861 CW53JC 11998038 Ki = 12 nM T44861 CQ39BY 12115602 IC50 = 4.4 nM T44861 C0BUN6 14058443 Ki = 80 nM T44861 C2BX8F 15297223 IC50 = 20 nM T44861 CE04YW 15297224 IC50 = 330 nM T44861 CFPW41 16007116 Ki > 8900 nM T44861 C9TU1O 16046126 IC50 > 1000 nM T44861 C86KBM 16123360 IC50 = 85 nM T44861 C68NYP 16123362 IC50 = 93 nM T44861 C8GTX1 16123589 IC50 = 3300 nM T44861 CV4CF9 16123704 IC50 = 3400 nM T44861 C8WNA0 16123709 IC50 = 1100 nM T44861 CR92JO 16124248 IC50 = 380 nM T44861 CP2M4O 16124345 IC50 = 88 nM T44861 CZF23I 16124479 IC50 = 316.23 nM T44861 C0H8UN 16730109 IC50 = 40000 nM T44861 C0WEX3 19966997 IC50 > 100000 nM T44861 C9AVK0 21113469 IC50 = 207 nM T44861 CS15LY 21672114 Ki = 0.41 nM T44861 CZ0X8J 22592015 IC50 > 315 nM T44861 CVR9K4 22907281 IC50 = 970 nM T44861 C0HRM6 22911602 IC50 = 300 nM T44861 CUN67H 23366085 IC50 = 112 nM T44861 CLG9Z8 23366090 IC50 = 5000 nM T44861 CW6OB1 23627212 IC50 = 17 nM T44861 CKYB29 23644745 IC50 = 50 nM T44861 CK73JS 24742033 Ki = 15 nM T44861 C2UOE0 24766030 IC50 = 1300 nM T44861 CJUK39 24770517 IC50 = 350 nM T44861 CY8X0J 24811794 Ki > 10000 nM T44861 CM28WD 24825721 IC50 = 51 nM T44861 CSW5V3 24865437 IC50 = 37 nM T44861 CPV6Y5 24866677 IC50 = 62 nM T44861 C36PKE 24992835 Ki = 255 nM T44861 CMP8Z9 24993483 Ki = 20 nM T44861 CH4RO0 24994728 Ki = 1300 nM T44861 C6E9WR 24995040 Ki = 255 nM T44861 CS3Q8B 24995659 Ki = 37 nM T44861 C2WXE1 24995663 Ki = 22 nM T44861 C1ONA4 24996161 IC50 = 44 nM T44861 CW38QS 25020248 IC50 = 1000 nM T44861 CY6I9E 25020250 IC50 = 881 nM T44861 CX1HL8 25032704 Ki > 8890 nM T44861 C0B7RT 25057409 IC50 > 10000 nM T44861 C6P1CX 25066843 IC50 = 26 nM T44861 CDO3X2 25113021 IC50 = 254 nM T44861 CBI73N 25113026 IC50 = 157 nM T44861 C1R0JL 25113028 IC50 = 53 nM T44861 C4KL8Q 25113038 IC50 = 124 nM T44861 CV58WZ 25113039 IC50 = 932 nM T44861 C8KI1Z 25113050 IC50 > 1000 nM T44861 CR0S2O 25195244 IC50 = 24 nM T44861 CTX60V 25195245 IC50 = 82 nM T44861 C92QDU 42611189 Ki = 240 nM T44861 CW24IK 42633780 Ki = 135 nM T44861 C75GFD 42633960 Ki = 184 nM T44861 CAO2T4 42634832 Ki = 584 nM T44861 CD5Z8U 44139091 Ki = 31.3 nM T44861 CAI56R 44139212 Ki = 46.4 nM T44861 CNX5R1 44139336 Ki = 11.6 nM T44861 CRD90G 44139337 Ki = 2.74 nM T44861 C4UMB7 44158300 Ki = 7.4 nM T44861 C4G5DI 44158301 Ki = 170 nM T44861 CLW80F 44160269 IC50 = 26 nM T44861 CLJ8U3 44186531 Ki = 590 nM T44861 CIX8V2 44251637 IC50 = 22 nM T44861 CGH06R 44251772 IC50 = 290 nM T44861 CP89VQ 44251773 IC50 = 81 nM T44861 C4FB3W 44251775 IC50 = 390 nM T44861 CZJO40 44251776 IC50 = 240 nM T44861 CB26IP 44251778 IC50 = 45 nM T44861 CM5LK7 44251903 IC50 = 240 nM T44861 CU93BX 44251904 IC50 = 200 nM T44861 CKZ3V2 44251905 IC50 = 15 nM T44861 CWUZ68 44251906 IC50 = 120 nM T44861 CX4AO2 44251907 IC50 = 56 nM T44861 CHW1Y9 44251908 IC50 = 28 nM T44861 CX23BG 44252049 IC50 = 29 nM T44861 C09WSD 44252050 IC50 = 33 nM T44861 C3VQ0G 44252052 IC50 = 77 nM T44861 C9JP5W 44252053 IC50 = 56 nM T44861 C7RFS9 44252054 IC50 = 180 nM T44861 C5GV6Y 44252348 IC50 = 930 nM T44861 C1S4EF 44252350 IC50 = 200 nM T44861 CNBS25 44252635 IC50 = 1600 nM T44861 CCV6J0 44252790 IC50 = 300 nM T44861 C9AP1D 44252942 IC50 = 34 nM T44861 C9QLC5 44253093 IC50 = 40 nM T44861 CWJ81C 44253525 IC50 = 72 nM T44861 CT6H2N 44253528 IC50 = 43 nM T44861 CLG7I2 44253664 IC50 = 67 nM T44861 C4JX5O 44253666 IC50 = 2.5 nM T44861 C4DIQ1 44253668 IC50 = 3.4 nM T44861 C9XVU8 44253795 IC50 = 250 nM T44861 CW4C0S 44253797 IC50 = 8 nM T44861 C5QFX6 44263382 IC50 = 47 nM T44861 C8RQU2 44263383 IC50 = 97 nM T44861 CZG81D 44263384 IC50 = 7.3 nM T44861 C6YRP1 44263385 IC50 = 794 nM T44861 CJHD91 44265316 Ki = 2500 nM T44861 C83QHW 44273476 IC50 > 100000 nM T44861 C3EFQ0 44273554 IC50 > 100000 nM T44861 CAJ48G 44273555 IC50 > 100000 nM T44861 C6VYU1 44273559 IC50 > 100000 nM T44861 C82YSI 44273595 IC50 > 100000 nM T44861 C0HG8U 44273619 IC50 > 100000 nM T44861 CMRX16 44273620 IC50 > 500000 nM T44861 C35TZW 44273659 IC50 > 100000 nM T44861 CG7M2O 44284055 Ki = 3 nM T44861 CQ13XB 44291629 Ki = 64.2 nM T44861 CERT91 44291669 Ki = 6.3 nM T44861 C1FZ6B 44294270 IC50 = 50 nM T44861 C6A9FK 44294365 IC50 = 5 nM T44861 C4HS3C 44294447 IC50 = 5 nM T44861 CFZ31C 44294493 IC50 = 20 nM T44861 C54GFD 44294623 IC50 = 5 nM T44861 CG89DS 44294661 IC50 = 100 nM T44861 CSHC96 44297347 IC50 = 2000 nM T44861 CYF8O6 44297594 IC50 = 300 nM T44861 CG1Z2B 44303442 IC50 = 30 nM T44861 CNJ63O 44303517 IC50 = 12 nM T44861 C8RJN7 44303745 IC50 = 220 nM T44861 CTM59P 44308069 IC50 = 5 nM T44861 CJ4WB9 44308383 IC50 = 6 nM T44861 C1N6SL 44308409 IC50 = 90 nM T44861 CO83HF 44308467 IC50 = 90 nM T44861 CYTA85 44308468 IC50 = 4000 nM T44861 C3M4UP 44308469 IC50 = 90 nM T44861 CY4K5F 44308490 IC50 = 32 nM T44861 C7AG9Y 44308609 IC50 = 4 nM T44861 CYN34A 44308610 IC50 = 20 nM T44861 C79WUE 44308611 IC50 = 6 nM T44861 CS63CK 44308612 IC50 = 20 nM T44861 C47BNR 44310732 IC50 = 4 nM T44861 C2ACB1 44310758 IC50 = 1 nM T44861 CXVB19 44310795 IC50 = 50 nM T44861 CD8OF2 44311036 IC50 = 5 nM T44861 C13TNU 44315122 IC50 = 100 nM T44861 C3YN1R 44315123 IC50 = 60 nM T44861 CPJ57U 44315124 IC50 = 40 nM T44861 C9HA8T 44315171 IC50 = 5 nM T44861 C2T3VN 44315184 IC50 = 340 nM T44861 C3SP0H 44315423 IC50 = 40 nM T44861 C8OAE9 44315457 IC50 = 35 nM T44861 C3JS6X 44315503 IC50 = 20 nM T44861 CEZ68T 44315545 IC50 = 100 nM T44861 CF61IT 44334334 IC50 = 1500 nM T44861 C3BFI4 44334443 IC50 = 610 nM T44861 CKD2B8 44337790 IC50 = 46000 nM T44861 COJ73E 44355185 Ki = 2.12 nM T44861 CIH03D 44366053 IC50 = 360 nM T44861 C9E2ZW 44373087 Ki = 0.8 nM T44861 C38PQK 44373108 Ki > 1000 nM T44861 C2B3PX 44373109 Ki = 0.8 nM T44861 CO28BT 44376126 Ki = 0.55 nM T44861 C8X0WA 44384580 Ki = 1370 nM T44861 CC95JU 44385548 IC50 = 420 nM T44861 CGQ57L 44386180 IC50 < 25 nM T44861 CI0Y5L 44386181 IC50 = 0.9 nM T44861 C1W6NC 44386587 IC50 = 5 nM T44861 C0PU3I 44386588 IC50 = 30 nM T44861 C3J6ZO 44386589 IC50 = 50 nM T44861 C4MZI9 44386931 IC50 = 21000 nM T44861 C6VJF9 44403780 Ki = 219 nM T44861 CETQ79 44427518 IC50 > 50000 nM T44861 COPG94 44427519 IC50 > 10000 nM T44861 CX6P0S 44449321 IC50 = 200 nM T44861 CUW91O 44449323 IC50 = 730 nM T44861 C3RHP2 44449448 IC50 = 310 nM T44861 CHZ8Y2 44449452 IC50 = 33000 nM T44861 CY87UN 44456923 Ki = 52.1 nM T44861 CW0T1S 44456924 Ki = 128 nM T44861 CS2CV1 44456938 Ki = 17.7 nM T44861 CCV59D 44473005 IC50 = 690 nM T44861 CX4V8F 44473006 IC50 = 260 nM T44861 CPZ9N7 44473007 IC50 = 94 nM T44861 CSA97D 44473008 IC50 = 120 nM T44861 C5WL1F 44473009 IC50 = 16 nM T44861 C6K7EH 44473010 IC50 = 27 nM T44861 CEG1S5 44473011 IC50 = 5.8 nM T44861 CQ02SK 44473012 IC50 = 18 nM T44861 C3MR8S 44473013 IC50 = 760 nM T44861 CXW6I3 44473014 IC50 = 62 nM T44861 C0Y5DZ 44473015 IC50 = 18 nM T44861 C46OMR 44473016 IC50 = 200 nM T44861 C5L0HD 44473017 IC50 = 310 nM T44861 CQG9E3 44473018 IC50 = 220 nM T44861 C97KBL 44473019 IC50 = 140 nM T44861 CP38JR 44473020 IC50 = 120 nM T44861 C8ZH6C 44473021 IC50 = 120 nM T44861 CLB89J 44473022 IC50 = 1300 nM T44861 CA03QZ 44473024 IC50 = 270 nM T44861 C73TDV 44473025 IC50 = 410 nM T44861 C02ZEH 44473028 IC50 = 120 nM T44861 C5QX6O 44511325 IC50 = 28 nM T44861 C3VRO9 44557921 IC50 > 10000 nM T44861 C8X1JW 44570801 IC50 = 51 nM T44861 CD9BY2 44570802 IC50 = 170 nM T44861 C5BNG9 44570803 IC50 = 250 nM T44861 CC58RY 44570848 IC50 = 410 nM T44861 CGWK29 44570849 IC50 = 27 nM T44861 CJY8S0 44570884 IC50 = 130 nM T44861 CYS8G0 44573871 IC50 = 2100 nM T44861 CTW62U 44573874 IC50 = 29 nM T44861 CEV7S0 44573875 IC50 = 30 nM T44861 CXK5I8 44573898 IC50 = 81 nM T44861 C3T1UP 44573899 IC50 = 980 nM T44861 CM9ZP7 44573901 IC50 = 280 nM T44861 COJ5C6 44573902 IC50 = 18 nM T44861 C7OGY2 44573903 IC50 = 110 nM T44861 CD65VM 44573904 IC50 = 41 nM T44861 CO18GC 44573905 IC50 = 160 nM T44861 C96NGB 44574269 IC50 = 350 nM T44861 C10YAL 44574270 IC50 = 69 nM T44861 C7C0FA 44574271 IC50 = 1400 nM T44861 C3LKQ1 44574272 IC50 = 63 nM T44861 C26CFS 44574273 IC50 = 85 nM T44861 CPG36C 44574310 IC50 = 210 nM T44861 C8OF9M 44574311 IC50 = 340 nM T44861 CAJY35 44574312 IC50 = 150 nM T44861 CF02XQ 44574313 IC50 = 130 nM T44861 C60ZRC 44578247 IC50 = 180 nM T44861 C6B1NX 44578248 IC50 = 100 nM T44861 C3YDK6 44578249 IC50 = 380 nM T44861 C7GDT1 44578680 IC50 = 450 nM T44861 C5AC1P 44578718 IC50 = 430 nM T44861 CL6I2W 44578719 IC50 = 340 nM T44861 C0E3VD 44578720 IC50 = 450 nM T44861 CSYM46 44578721 IC50 = 4100 nM T44861 C8TUL6 44578755 IC50 = 200 nM T44861 CT0WO1 44578756 IC50 = 73 nM T44861 CK23LX 44578757 IC50 = 67 nM T44861 C8AD1R 44578758 IC50 = 2100 nM T44861 C01KPH 44578813 IC50 = 250 nM T44861 C67MLJ 44578814 IC50 = 500 nM T44861 CCY0X5 44578815 IC50 = 500 nM T44861 C0KM7V 44578816 IC50 = 1800 nM T44861 CMG72K 44578839 IC50 = 790 nM T44861 C34SOM 44578840 IC50 = 420 nM T44861 C98BRO 44578841 IC50 = 330 nM T44861 CRNT03 44578842 IC50 = 1800 nM T44861 CI7MN3 44621943 Ki = 526 nM T44861 C1V6TC 44622679 Ki = 722 nM T44861 CPTY61 44626360 IC50 = 4.3 nM T44861 C06WDZ 45107770 Ki = 89 nM T44861 C7BQ2T 45108044 Ki = 151 nM T44861 C46FDT 45108081 Ki = 132 nM T44861 C16IEQ 45108117 Ki = 81 nM T44861 C8GFI2 45108120 Ki = 336 nM T44861 CC95PQ 45375865 IC50 = 18 nM T44861 CEOQ27 45375866 IC50 = 65 nM T44861 C9VJH6 45484979 IC50 = 1100 nM T44861 C0Y1ZH 45484983 IC50 = 41 nM T44861 CM6ZH3 45484989 IC50 = 880 nM T44861 C1T3JI 45484990 IC50 = 140 nM T44861 C4P3XB 45484994 IC50 = 25 nM T44861 CR52GN 45485014 IC50 = 10000 nM T44861 CXA0O7 45485015 IC50 = 670 nM T44861 C84AUV 45485016 IC50 = 81 nM T44861 CG97AV 45485017 IC50 = 350 nM T44861 C8BQ5R 45485037 IC50 = 420 nM T44861 C8M5XT 45485046 IC50 = 64000 nM T44861 C3NYJ6 45485051 IC50 = 800 nM T44861 CA5VN0 45485052 IC50 = 110 nM T44861 C3RDZ0 45485058 IC50 = 620 nM T44861 CM93TU 45485059 IC50 = 62 nM T44861 CTK16A 45485067 IC50 = 1400 nM T44861 CNPW65 45485068 IC50 = 150 nM T44861 CEY2C0 45485076 IC50 = 34 nM T44861 C2S1PV 45485082 IC50 = 3500 nM T44861 C5S8MA 45485083 IC50 = 53 nM T44861 CSA2U3 45485596 IC50 = 57 nM T44861 CF8U6I 45485719 IC50 = 10 nM T44861 CX7I1G 45485730 IC50 = 154 nM T44861 CP1TD8 45485731 IC50 = 25 nM T44861 CSC38R 45485732 IC50 = 44 nM T44861 C3ZHD5 45485733 IC50 = 13 nM T44861 CJ94MU 45485734 IC50 = 21 nM T44861 C3QJ2U 45485738 IC50 = 43 nM T44861 C6LT4C 45485739 IC50 = 121 nM T44861 C2P3WG 45485740 IC50 = 16 nM T44861 CS1R6E 45485748 IC50 = 16 nM T44861 CZYD36 45485761 IC50 = 5.2 nM T44861 C2B5JI 45485762 IC50 = 20 nM T44861 CUJ6X4 45485765 IC50 = 138 nM T44861 CS1K2D 45485766 IC50 = 149 nM T44861 C03NFZ 45485774 IC50 = 110 nM T44861 C6O5BP 45485797 IC50 = 9.9 nM T44861 CD3GS6 45487537 IC50 = 36 nM T44861 C0ATH1 45487554 IC50 = 86 nM T44861 CTR3P4 45487555 IC50 = 94 nM T44861 CHT58B 45487559 IC50 = 250 nM T44861 CFV38T 45487561 IC50 = 390 nM T44861 CW3F7U 45487562 IC50 = 300 nM T44861 C5X8YN 45487570 IC50 = 58 nM T44861 CU2J5S 45487571 IC50 = 25 nM T44861 CA0CB9 45487572 IC50 = 190 nM T44861 CO0X4N 45487573 IC50 = 8.2 nM T44861 C6AHT9 45487574 IC50 = 14 nM T44861 CE3F2I 45487575 IC50 = 18 nM T44861 CI24NY 45487588 IC50 = 2400 nM T44861 CRJ5X1 45487595 IC50 = 25 nM T44861 CL3K8H 45487596 IC50 = 22 nM T44861 C8HN1Y 45487597 IC50 = 50 nM T44861 CCV15K 45487611 IC50 = 70 nM T44861 C76RIH 45487622 IC50 = 84 nM T44861 C5CLP8 45487627 IC50 = 9.7 nM T44861 CW42YX 45487634 IC50 = 45 nM T44861 CY3HW5 46224684 IC50 = 860 nM T44861 C6SL3O 46227444 IC50 = 2000 nM T44861 C8UJT1 46227519 IC50 = 250 nM T44861 CQW97N 46846072 IC50 = 29 nM T44861 CLS29B 46872626 IC50 > 10000 nM T44861 CKR46X 46879514 IC50 = 140 nM T44861 CCS06U 46879515 IC50 = 450 nM T44861 CQ1XO5 46879516 IC50 = 20000 nM T44861 CB6DH0 46879555 IC50 = 114 nM T44861 CF04OQ 46879556 IC50 = 1300 nM T44861 CP3K1R 46879557 IC50 = 3300 nM T44861 CN90TO 46879558 IC50 = 51000 nM T44861 C7H9NW 46879602 IC50 = 9400 nM T44861 CWJH34 46879604 IC50 = 120 nM T44861 CNUT90 46879605 IC50 = 390 nM T44861 CR14YD 46879645 IC50 = 850 nM T44861 C8DH4B 46879687 IC50 = 2000 nM T44861 CU51HD 46879688 IC50 = 4400 nM T44861 CJV29C 46879689 IC50 = 7100 nM T44861 CZXU95 46879733 IC50 = 21000 nM T44861 CS0NZ6 46879734 IC50 = 320 nM T44861 CRV8H5 46879735 IC50 = 94 nM T44861 C0AW5F 46879777 IC50 = 110 nM T44861 CL6GX0 46879778 IC50 = 97 nM T44861 CLC24S 46881462 IC50 = 24 nM T44861 CN04PB 46881504 IC50 = 96 nM T44861 COZS08 46881505 IC50 = 68 nM T44861 CARX78 46881506 IC50 = 240 nM T44861 CC9F7R 46881553 IC50 = 180 nM T44861 C8DS7P 46881554 IC50 = 51 nM T44861 CWP05I 46881555 IC50 = 16 nM T44861 C2LF8C 46881556 IC50 = 45 nM T44861 CRVO58 46881593 IC50 = 75 nM T44861 CF5M1N 46881594 IC50 = 45 nM T44861 CRC2J7 46881595 IC50 = 85 nM T44861 C4XBI1 46881640 IC50 = 53 nM T44861 CP4F9B 46881641 IC50 = 41 nM T44861 C5W8KJ 46881678 IC50 = 770 nM T44861 C8DBP9 46881679 IC50 = 76 nM T44861 C0TE7Y 46881680 IC50 = 55 nM T44861 C0NI6L 46881681 IC50 = 150 nM T44861 CVG0L2 46881723 IC50 = 130 nM T44861 CKG50T 46881724 IC50 = 36 nM T44861 CQN09T 46881725 IC50 = 61 nM T44861 CW37OB 46881726 IC50 = 61 nM T44861 C9YGL1 46881774 IC50 = 18 nM T44861 CH4UA0 46881775 IC50 = 43 nM T44861 CEAZ53 46881776 IC50 = 11 nM T44861 C1IGH5 46881777 IC50 = 90 nM T44861 C2O8RZ 46886323 IC50 > 1000 nM T44861 CVJ4K0 46899547 IC50 = 963 nM T44861 C2B8IC 46899551 IC50 = 1000 nM T44861 CSV5B9 46901859 IC50 = 20 nM T44861 C7YJ2X 46901862 IC50 = 31 nM T44861 C9L3XR 49838879 IC50 > 40000 nM T44861 C96RSQ 49864366 Ki = 27000 nM T44861 CCL6T7 49870878 IC50 = 25118.86 nM T44861 CHP06V 52948258 Ki = 9.8 nM T44861 CR93CL 53308750 Ki = 18 nM T44861 CD4H3S 53354074 Ki = 16 nM T44861 CB32QT 53354075 Ki = 242 nM T44861 C8AB5U 53354478 Ki < 10 nM T44861 C8NA4L 53384644 IC50 = 15000 nM T44861 CUY9G2 53473663 IC50 = 27 nM T44861 CGQ7F8 53473746 IC50 = 3.2 nM T44861 CI1ZG3 53473747 IC50 = 0.6 nM T44861 C67JHW 53473748 IC50 = 1.2 nM T44861 C7EW6O 53473749 IC50 = 4.1 nM T44861 CPH34R 53473750 IC50 = 12 nM T44861 CWH1D4 53473825 IC50 > 316 nM T44861 CM8K2V 53473826 IC50 = 6.3 nM T44861 C9A8HG 53473827 IC50 = 224 nM T44861 C3A8OT 53473828 IC50 = 52 nM T44861 CLX31Q 53473829 IC50 = 93 nM T44861 C8Y9RE 53473918 IC50 = 2.5 nM T44861 C1XFN0 53473919 IC50 = 8.2 nM T44861 CN34UO 53473920 IC50 = 6.2 nM T44861 C2RE5M 53473921 IC50 = 0.1 nM T44861 C9ZUL0 53473922 IC50 = 5.7 nM T44861 CG6FD5 53474007 IC50 = 2.7 nM T44861 C0Q7JS 53474008 IC50 = 25 nM T44861 C31WZB 53474009 IC50 = 1 nM T44861 CJF1M2 53630890 IC50 = 214 nM T44861 CCM71K 54669828 Ki = 87 nM T44861 CNB76L 56643505 IC50 = 8 nM T44861 CYB2X7 56841025 EC50 = 4.7 nM T44861 CE25GK 57392822 EC50 = 25230 nM T44861 CP0L8E 57690510 Ki = 30 nM T44861 CS9E2N 57690531 Ki = 87 nM T44861 C2J9WL 57690545 Ki < 10 nM T44861 CQ0OR2 57690846 Ki = 80 nM T44861 CSP2I8 57690850 Ki > 2000 nM T44861 CAU57Q 57969602 Ki = 60 nM T44861 C1LZI4 57969746 Ki = 392 nM T44861 COH41P 58325285 IC50 = 18 nM T44861 CU38PN 58367655 Ki = 116 nM T44861 CJ6ZT2 59332810 IC50 = 294 nM T44861 CNL04P 60155126 Ki = 3.3 nM T44861 C56PUM 60155209 Ki = 0.46 nM T44861 CV63UL 67240318 IC50 > 10000 nM T44861 CJM08K 67949700 Ki = 358 nM T44861 CJX61W 67949768 Ki > 1250 nM T44861 C2PWR3 67949769 Ki = 130 nM T44861 CJ1CK8 67949771 Ki > 1250 nM T44861 CA43IM 67949780 Ki = 792 nM T44861 CWZ6B3 67949822 Ki = 131 nM T44861 C8KR4F 67949825 Ki = 480 nM T44861 C45HUR 68027012 EC50 = 5.3 nM T44861 CVR5Z6 68027063 EC50 = 4.5 nM T44861 C6Y7NH 68036615 EC50 = 3.3 nM T44861 CH87DV 68036617 EC50 = 19.8 nM T44861 CT37OB 68036619 EC50 = 156 nM T44861 C06LGW 68036621 EC50 = 13.4 nM T44861 CH90KJ 68036622 EC50 = 8 nM T44861 C5WJC7 68036669 EC50 = 4.2 nM T44861 C8F4HT 68036689 EC50 = 2.9 nM T44861 CMN0F3 68036705 EC50 = 25.7 nM T44861 CN1JR7 68036706 EC50 = 13.1 nM T44861 CF39DV 68596931 IC50 = 214 nM T44861 C9XLB3 68597337 IC50 = 63 nM T44861 CMQ58W 68597501 IC50 = 635 nM T44861 CEZU83 68611347 IC50 = 703 nM T44861 CJ8G3H 68682755 IC50 = 254 nM T44861 CJGH31 70285522 IC50 > 1000 nM T44861 CPZ4F6 71451107 IC50 > 1000 nM T44861 C5RKX0 71452928 IC50 = 102 nM T44861 CKT60L 71455860 Ki = 7.9 nM T44861 CLZ67D 71456431 IC50 > 1000 nM T44861 CS89CL 71456432 IC50 = 371 nM T44861 CPIH21 71460129 IC50 = 221 nM T44861 C69NCX 71461845 IC50 > 1000 nM T44861 C9QB5V 71461846 IC50 > 1000 nM T44861 C6O8KG 71461847 IC50 = 386 nM T44861 C07RPM 71583135 Ki = 57 nM T44861 C97WFL 71583136 Ki > 1250 nM T44861 C07HUA 71583137 Ki = 120 nM T44861 CR2P7K 71583245 Ki > 1250 nM T44861 CIQK36 71583246 Ki = 547 nM T44861 C4MOE6 71583247 Ki = 957 nM T44861 C3VE2F 71658602 Ki = 690 nM T44861 C4GS3M 71658603 Ki = 36 nM T44861 C3VO6X 71658604 Ki = 3.5 nM T44861 CQIL32 71658605 Ki = 4.1 nM T44861 CG8W1H 71658606 Ki = 6.9 nM T44861 CF1A2P 71658736 Ki = 1.3 nM T44861 CBPU84 71658737 Ki = 4.6 nM T44861 C31ZKG 71658738 Ki = 9.7 nM T44861 CU60JG 71718528 IC50 = 42000 nM T44861 CV70GZ 71728100 Ki = 0.32 nM T44861 CK2DT6 72737674 EC50 = 5.2 nM T44861 CI0P4Y 73347739 EC50 = 10.6 nM T44861 C53IUO 73349295 EC50 = 6.1 nM T44861 CAS36F 73350862 EC50 = 5.3 nM T44861 C7Q0AD 76286479 IC50 = 330 nM T44861 CZF0N7 76287389 IC50 = 470 nM T44861 C28STM 76287526 IC50 = 750 nM T44861 C26HPB 76310178 EC50 = 2.5 nM T44861 C7YN4K 76313879 EC50 = 3.8 nM T44861 C3TN6S 76324778 EC50 = 988 nM T44861 C1B7EA 76324779 EC50 = 3.7 nM T44861 CICS73 76331997 EC50 > 10000 nM T44861 CF5P2Z 76331998 EC50 = 10.8 nM T44861 C0Y8ZK 91933875 IC50 > 10 nM T44861 C8Z6KW 101873991 Ki = 18 nM T44861 C9D7RT 101874012 Ki = 28 nM T44861 CLX42P 101874014 Ki = 2.7 nM T44861 CS6YH1 101874015 Ki = 2.8 nM T44861 CRYU45 101874016 Ki = 1.3 nM T44861 C2GZ8E 101874017 Ki = 7.6 nM T44861 CK1O6M 101874018 Ki > 250 nM T44861 CG4JB9 122194654 IC50 = 39900 nM T44861 C2VQW1 134817176 EC50 = 8030 nM T44861 C2KFH7 135398497 Ki = 318 nM T44861 CS4OW8 135400873 Ki = 320 nM T44861 CSB0M9 135494223 EC50 = 14970 nM T44861 CRJ45X 135589980 IC50 > 50000 nM T44861 CFAD48 135611170 Ki = 480 nM T44861 C0J3BN 135678111 IC50 > 50000 nM T44861 C1XQY2 135923992 EC50 = 11550 nM T44861 CC65KF 136042192 EC50 = 21640 nM T44861 C26ESH 136060555 IC50 > 50000 nM T44861 CJ7KN6 136250327 Ki < 10 nM T44861 C12UXT 137640959 IC50 > 316 nM T44861 CH15QZ 137643717 IC50 = 230 nM T44861 CUG6N7 137660315 IC50 = 39 nM T44861 C6QA5D 137661222 IC50 = 284 nM T44861 C6VB3O 145925651 IC50 >= 5000 nM T44861 CEV2U7 145967191 Ki = 1000 nM T44861 C2MD1Q 155513187 IC50 > 10000 nM T44861 CM42JV 155519536 Ki = 4 nM T44861 CSR65F 155539817 Ki = 1200 nM T44861 CK52UC 155542191 Ki = 12 nM T44861 CSZ98D 155544487 Ki = 3.4 nM T44861 CBO72N 155547084 Ki = 1.9 nM T44861 C41LAG 155547541 Ki = 7.9 nM T44861 CE73YI 155548741 Ki = 3.3 nM T44861 CBQ59W 155550296 Ki = 5.1 nM T44861 C0XVI4 155551436 Ki = 5.9 nM T44861 CLQ07Y 155554050 Ki = 3.6 nM T44861 CDT92F 155560040 Ki = 9.1 nM T44861 C85GOK 155560969 Ki = 880 nM T44861 C8T6GL 155561087 Ki = 4.4 nM T44861 CU34OH 155567589 Ki = 542 nM T44861 D00ERW 44444843 Ki > 8889 nM T44861 D00HVA 11624601 Ki > 8900 nM T44861 D02KPV 37783 Ki = 0.8 nM T44861 D02XHC 448912 IC50 > 100000 nM T44861 D04AXH 11574614 Ki = 216 nM T44861 D05SLL 44186619 Ki = 529 nM T44861 D06ZCX 10455969 IC50 = 690 nM T44861 D07ANB 148879 EC50 = 16150 nM T44861 D07OAT 456214 IC50 > 100000 nM T44861 D08JPU 3501 IC50 = 446 nM T44861 D09XIL 11396738 IC50 > 125000 nM T44861 D0CM6T 11314340 Ki = 360 nM T44861 D0D6DH 10125830 IC50 > 50000 nM T44861 D0J4NI 44186618 Ki = 915 nM T44861 D0K5ZY 105000 Ki = 8.2 nM T44861 D0Q3NG 11715520 Ki > 8900 nM T44861 D0S7IE 11658882 Ki > 8900 nM T44861 D0TO6S 2396 IC50 = 8.7 nM T44861 D0U9YY 45485012 IC50 = 240 nM T97719 D03ZBT 11626560 IC50 > 10000 nM T97719 D04LVK 57379345 IC50 = 3360 nM T97719 D05NUH 54758501 IC50 = 1 nM T97719 D09KTS 24821094 IC50 = 0.1 nM T97719 D09PQZ 71226662 IC50 = 3.1 nM T97719 D0E6XR 3062316 IC50 = 1.3 nM T97719 D0OB0F 5328940 IC50 = 2.5 nM T97719 D0R3JB 4212 IC50 = 1000 nM T97719 D02TUL 118115473 IC50 = 607 nM T97719 D03LWG 53235510 IC50 > 10000 nM T97719 D04BFC 59174488 IC50 = 0.6 nM T97719 D07EHV 44814409 IC50 > 10000 nM T97719 D07HPJ 11476171 IC50 = 7600 nM T97719 D08AOZ 86582336 IC50 = 0.5 nM T97719 D0E3TC 44259 IC50 = 13.38 nM T97719 D0FD6D 11751922 IC50 = 93 nM T97719 D0G5XV 135565884 IC50 = 0.3 nM T97719 D0H0KH 54755438 IC50 = 5.2 nM T97719 D0O6WV 24794418 IC50 > 2000 nM T97719 D0QX8X 71479709 IC50 = 61 nM T97719 D0U7KH 86567195 Ki = 0.91 nM T97719 D0UT4W 135905454 IC50 = 0.63 nM T97719 D0YB3W 156414 IC50 = 185 nM T97719 D0Q1BE 72188716 IC50 = 6.5 nM T97719 D03FUO 25234918 IC50 = 14 nM T97719 D0T3ME 156422 IC50 > 30000 nM T97719 CR98MZ 613528 IC50 = 4100 nM T97719 C0ZI1F 2756534 IC50 = 15100 nM T97719 CI0P2J 2814562 IC50 = 3500 nM T97719 CXW3U6 3031415 IC50 > 6000 nM T97719 CPXK25 5793057 IC50 = 5150 nM T97719 CB7WK3 5938113 IC50 = 6700 nM T97719 CP0XI6 6603792 IC50 = 310 nM T97719 CM5Z8X 9869943 IC50 = 0.4 nM T97719 CSGD16 10246246 IC50 > 7000 nM T97719 C7SFI1 10296883 IC50 > 10000 nM T97719 CJ7U4I 11161778 IC50 = 23000 nM T97719 CW5C9X 11186250 IC50 = 1258.93 nM T97719 CRC86K 11397050 IC50 = 400 nM T97719 CM21YJ 11453049 IC50 = 1584.89 nM T97719 C7HMO6 11526786 IC50 > 10000 nM T97719 CACS26 11561968 Ki > 2000 nM T97719 CJ9KN7 11683817 IC50 > 10000 nM T97719 CU0E8O 11690457 Ki > 10000 nM T97719 C45EWD 11723489 IC50 > 7000 nM T97719 CP7AH3 11755812 IC50 = 7800 nM T97719 CS36BH 11843159 IC50 = 100 nM T97719 C2IS9W 11851477 IC50 = 150 nM T97719 CJXK96 11851580 IC50 = 60 nM T97719 CCN9L1 11851680 IC50 = 230 nM T97719 CJ6S2Q 11851879 IC50 = 30 nM T97719 C0FGK3 11852095 IC50 = 130 nM T97719 CF4S5D 11852469 IC50 = 21 nM T97719 CHR92S 11858109 IC50 = 27 nM T97719 C9RQN8 15950748 IC50 = 3423 nM T97719 C09OWB 16015442 IC50 = 1091 nM T97719 CKR57M 16086104 IC50 = 3330 nM T97719 C16NRY 16086114 IC50 = 545 nM T97719 CQG45C 16109001 IC50 = 25000 nM T97719 C5VPH9 16129448 IC50 = 4950 nM T97719 CL9BQ6 17748275 IC50 = 25000 nM T97719 CWH37T 17758574 IC50 > 10000 nM T97719 CAFW78 18450761 IC50 = 1954 nM T97719 C6BA1Y 18450866 IC50 = 767.5 nM T97719 CA61QF 21083895 IC50 = 17000 nM T97719 CFP37A 22347110 IC50 = 8.2 nM T97719 C6JV7W 23400934 IC50 > 7000 nM T97719 CD5S7O 23401001 IC50 > 7000 nM T97719 CK5N6B 23657635 IC50 = 97 nM T97719 CIZ4V1 24756997 IC50 = 9 nM T97719 C7YG1N 24759534 IC50 = 290 nM T97719 CQNP54 24764449 IC50 = 1000 nM T97719 C4Z9CN 24769780 IC50 = 126 nM T97719 CJUK39 24770517 IC50 > 10000 nM T97719 C9PA0M 24807809 IC50 > 10000 nM T97719 C9F1AO 24821023 IC50 = 0.5 nM T97719 CBW43O 24821811 IC50 = 20 nM T97719 CI5MQ1 24821812 IC50 = 0.58 nM T97719 CY48ZA 24821879 IC50 = 0.72 nM T97719 CY8L7E 24896769 IC50 > 10000 nM T97719 CIM4Q1 24901165 IC50 = 875 nM T97719 CFI7S2 24936376 IC50 = 13 nM T97719 C4KG6Z 24968331 IC50 = 42 nM T97719 CD5HQ0 24969301 IC50 > 10000 nM T97719 CD69RK 25097993 IC50 > 10000 nM T97719 C36FXD 25138012 IC50 = 9 nM T97719 CP6N4G 25138050 IC50 = 69 nM T97719 CSO82D 25154877 Ki = 0.25 nM T97719 CJL25F 25169253 IC50 = 5 nM T97719 C9Y0JV 25206375 IC50 = 8 nM T97719 CLH0V2 25234052 IC50 = 61 nM T97719 C1RU9T 25234054 IC50 = 1400 nM T97719 CKC10Q 25234136 IC50 = 88 nM T97719 C4D6UF 25234139 IC50 = 5 nM T97719 C2TPV7 25234524 IC50 = 6 nM T97719 C4MAC1 25234917 IC50 = 20 nM T97719 C6PQ7E 25234978 IC50 = 6 nM T97719 CNI4C8 25235043 IC50 = 3 nM T97719 C67VMP 25235106 IC50 = 20 nM T97719 C21DQU 25235170 IC50 = 5.9 nM T97719 CDU9Q6 25235171 IC50 = 9 nM T97719 CQD83X 25235172 IC50 = 14 nM T97719 C3L6ER 25235173 IC50 = 15 nM T97719 CZ64OU 25235174 IC50 = 9 nM T97719 CRO8T9 25263033 Ki = 125 nM T97719 CN5E0F 25263283 IC50 = 14000 nM T97719 CS2EW5 25264176 IC50 = 13 nM T97719 CK31XP 44182938 IC50 = 280 nM T97719 CB53SU 44182939 IC50 = 1600 nM T97719 CA98KR 44432441 IC50 > 22000 nM T97719 C6GP5Z 44548488 IC50 = 200 nM T97719 CLXZ05 44554064 IC50 = 38 nM T97719 C3VRO9 44557921 IC50 > 10000 nM T97719 C3XTA7 44562721 Ki = 78 nM T97719 C3HW7L 44570553 IC50 > 30000 nM T97719 C17PVE 44570554 IC50 > 30000 nM T97719 CLOY92 44570599 IC50 = 7000 nM T97719 CK06LT 44570600 IC50 > 30000 nM T97719 CMO3R5 44602494 IC50 = 30 nM T97719 C70VXL 44624435 IC50 = 144 nM T97719 CX0U3N 46220516 IC50 = 2 nM T97719 CB7WM8 46222818 IC50 = 10 nM T97719 C8JM5X 46223487 IC50 = 103 nM T97719 C0YTF8 46223725 IC50 = 132 nM T97719 CG71EF 46832441 IC50 = 327 nM T97719 C1LNX9 46832443 IC50 = 436 nM T97719 CH0JZ8 46833813 IC50 = 19 nM T97719 CD17VE 46833814 IC50 = 12 nM T97719 C9NCS8 46833815 IC50 = 11 nM T97719 C7H4YM 46865419 IC50 > 10000 nM T97719 CLS29B 46872626 IC50 > 10000 nM T97719 CZK6C2 46894111 IC50 = 8 nM T97719 CRB9E6 46908028 IC50 = 400 nM T97719 CF3Y7V 46908220 IC50 = 3 nM T97719 CKC0D5 46908221 IC50 = 2 nM T97719 CIG9W1 46908418 IC50 = 40 nM T97719 C9U6PT 46908706 IC50 = 50 nM T97719 CX9CT2 46909487 IC50 = 4 nM T97719 C9PAT7 46927672 IC50 = 10 nM T97719 C60GAV 46929544 IC50 > 8000 nM T97719 CP34VL 46929748 IC50 > 1000 nM T97719 CJ2E9Q 46929857 IC50 > 25000 nM T97719 CX65UM 49787738 IC50 = 2 nM T97719 C9L3XR 49838879 IC50 > 15000 nM T97719 CL4R0T 50925568 IC50 = 20 nM T97719 CI2VR3 51000608 IC50 = 4900 nM T97719 CDU90A 51000695 IC50 = 45000 nM T97719 C4P6MB 51000778 IC50 = 800 nM T97719 CWAX19 51000932 IC50 = 120 nM T97719 CR1W4B 51000933 IC50 = 1800 nM T97719 C5J4ZC 51000934 IC50 = 2300 nM T97719 CG8RL9 51000936 IC50 = 2700 nM T97719 CV0YT2 51000937 IC50 = 3200 nM T97719 CWOS84 51001012 IC50 > 10000 nM T97719 CO8UM9 51001094 IC50 = 200 nM T97719 CRNH80 51001177 IC50 = 100 nM T97719 C4E3LI 51001515 IC50 = 19000 nM T97719 C93AED 51001516 IC50 = 44000 nM T97719 CEQN27 52936621 Ki > 1000 nM T97719 C2W9OA 53324451 IC50 > 10000 nM T97719 C8ZRE3 53356518 IC50 = 8 nM T97719 C8NA4L 53384644 IC50 > 30000 nM T97719 CRD4Z6 54596323 IC50 = 8 nM T97719 CG1RK0 54596453 Ki = 0.69 nM T97719 CNH42M 54596723 Ki = 1.28 nM T97719 CM8JX1 56604907 IC50 = 10 nM T97719 CD3P6C 56644522 IC50 = 651.95 nM T97719 C6AN2Z 56656450 IC50 < 1 nM T97719 CJBL48 56925034 IC50 = 15 nM T97719 C18CKJ 56928445 IC50 = 3 nM T97719 C3KY5Z 56928861 IC50 = 3 nM T97719 CQGH97 57391046 IC50 = 13.2 nM T97719 C8GQ9H 57391143 IC50 = 1.55 nM T97719 CSU96R 57391144 IC50 = 76.5 nM T97719 C7OQ2B 57391145 IC50 = 13 nM T97719 C3X1ZN 57392910 IC50 = 3.33 nM T97719 COC5U3 57392911 IC50 = 1.89 nM T97719 CN03CZ 57392994 IC50 = 0.884 nM T97719 C2DRH3 57392995 IC50 = 19.1 nM T97719 CE1A9V 57394653 IC50 = 0.7 nM T97719 CIQH60 57394654 IC50 = 6.76 nM T97719 CD5Z9R 57394655 IC50 = 4.83 nM T97719 CNV76Z 57394656 IC50 = 2.6 nM T97719 CO34BP 57394657 IC50 = 40 nM T97719 C8W6IG 57395117 IC50 > 30000 nM T97719 CH2PZ8 57396405 IC50 = 6.58 nM T97719 CN8I2E 57396406 IC50 = 1220 nM T97719 C3NG0U 57396491 IC50 = 0.847 nM T97719 CNC84H 57396492 IC50 = 45.3 nM T97719 COG41M 57398104 IC50 = 7.56 nM T97719 C83EBV 57398105 IC50 = 60.6 nM T97719 CL78SU 57398205 IC50 = 12.2 nM T97719 CVRX72 57398206 IC50 = 9.53 nM T97719 C05PSA 57398207 IC50 = 72 nM T97719 CBK0C1 57399762 IC50 = 10.3 nM T97719 C4CQR0 57399857 IC50 = 5.51 nM T97719 COC32E 57401532 IC50 = 10.4 nM T97719 C7Z4PU 57401624 IC50 = 16.8 nM T97719 C7M2NU 57401629 IC50 = 1.82 nM T97719 CET8G9 57401630 IC50 = 5.35 nM T97719 C1CJ3Y 57401631 IC50 = 5.03 nM T97719 CCT87N 57401632 IC50 = 9.53 nM T97719 CDS7G4 57401633 IC50 = 670 nM T97719 C5THG9 57401721 IC50 = 2.52 nM T97719 C6LWX8 57401722 IC50 = 3.99 nM T97719 CU1C9S 57401723 IC50 = 4290 nM T97719 CZ4UR3 57403361 IC50 = 2.96 nM T97719 CY1Z7M 57403363 IC50 = 283 nM T97719 CG0Y3M 57403447 IC50 = 0.847 nM T97719 C3YGA0 57424138 IC50 = 3700 nM T97719 CG0O6Y 57473392 IC50 = 190 nM T97719 CNU76E 58043734 IC50 = 6 nM T97719 CD10RZ 58043863 IC50 = 81 nM T97719 C9JOQ3 58044026 IC50 = 4 nM T97719 C6J7QV 58044116 IC50 = 4 nM T97719 CY7N4D 58044297 IC50 = 1 nM T97719 CQEN24 58044306 IC50 = 2 nM T97719 CCF7Z0 58540029 IC50 = 4 nM T97719 C4KJL2 58540036 IC50 = 11 nM T97719 CPIF95 58540060 IC50 = 4 nM T97719 CMDI08 58540134 IC50 = 1 nM T97719 C68GRX 58540298 IC50 = 20 nM T97719 CR7WI1 58540323 IC50 = 4 nM T97719 CV13QY 58540422 IC50 = 3 nM T97719 CQ8VU9 58728932 IC50 = 8.9 nM T97719 C0EOY8 58729072 IC50 = 50 nM T97719 CCP4Z1 58729084 IC50 = 50 nM T97719 C94EVL 58729093 IC50 = 230 nM T97719 C1SI3L 59174579 IC50 < 1 nM T97719 COT79B 59216480 IC50 = 60 nM T97719 CT3EW2 59292007 IC50 > 1000 nM T97719 C2V9LI 59375017 IC50 = 9 nM T97719 C1L4FX 59375068 IC50 = 29 nM T97719 CBY4S3 59375142 IC50 = 11 nM T97719 CZ3TG1 59375154 IC50 = 16 nM T97719 CXJ63M 59603829 IC50 = 360 nM T97719 CQEU96 59603842 IC50 < 1 nM T97719 C1MR8Q 60097495 IC50 > 1000 nM T97719 CSZ6I5 66556035 IC50 = 251.19 nM T97719 C3ER5W 66601644 IC50 = 2 nM T97719 CD0LJ6 66604359 IC50 = 461 nM T97719 CT4RU2 66604890 IC50 = 189 nM T97719 C0JS8O 66604914 IC50 = 110 nM T97719 C0EVU7 66605043 IC50 = 379 nM T97719 CGS8J2 66605151 IC50 = 404 nM T97719 CCWU74 66605322 IC50 = 360 nM T97719 CN5BR8 66605844 IC50 = 308 nM T97719 CDES25 66606401 IC50 = 812 nM T97719 C9O2RZ 66895259 IC50 = 110 nM T97719 CSR94E 66895407 IC50 = 270 nM T97719 CQN0H3 66895621 IC50 = 70 nM T97719 CN7F2G 66926889 IC50 = 1 nM T97719 CW9RF7 67016212 Ki = 0.35 nM T97719 CKRX65 67016282 IC50 = 16700 nM T97719 CY9SL3 67016323 IC50 = 2600 nM T97719 C4U3XP 67016524 IC50 = 3 nM T97719 C1HSE0 67035086 IC50 = 580 nM T97719 CWI6K5 67035106 IC50 > 10000 nM T97719 C38RGB 67035556 IC50 > 10000 nM T97719 C37NKO 67129970 IC50 > 10000 nM T97719 CK80LJ 67130050 IC50 > 10000 nM T97719 CV63UL 67240318 IC50 > 10000 nM T97719 CR7DC4 67969461 IC50 < 100 nM T97719 CAF36T 67972044 IC50 = 9 nM T97719 C78QYC 67972152 IC50 < 100 nM T97719 C56FMK 67986337 IC50 < 100 nM T97719 CE4SM9 67986343 IC50 = 140 nM T97719 C7ARX2 67986346 IC50 = 460 nM T97719 CVZE42 67986349 IC50 = 550 nM T97719 C8C4ZF 67986352 IC50 = 400 nM T97719 CP7BO8 67986356 IC50 = 1200 nM T97719 CZY09U 67986357 IC50 = 1300 nM T97719 CZJ40Q 67986358 IC50 = 500 nM T97719 CLQ91B 67986410 IC50 > 10000 nM T97719 CLUR72 67986417 IC50 > 20000 nM T97719 CZNS75 68051325 IC50 < 100 nM T97719 C8I7GC 68293638 IC50 > 10000 nM T97719 CD56XK 68293660 IC50 > 10000 nM T97719 C7GRV2 68755406 IC50 > 10000 nM T97719 C5DGR9 69036886 IC50 = 1879 nM T97719 C3GTU1 69762142 IC50 > 10000 nM T97719 CY57QX 70647721 IC50 = 34 nM T97719 CD3A0B 70647727 IC50 = 3 nM T97719 C7VJ6A 70647728 IC50 = 2.6 nM T97719 C6E8DC 71092932 IC50 = 8600 nM T97719 CBKF84 71222614 IC50 = 0.3 nM T97719 C82IYH 71222927 IC50 = 10.7 nM T97719 CLIH32 71226367 IC50 = 0.3 nM T97719 CE4Y8J 71226521 IC50 = 11 nM T97719 CT4P8G 71226707 IC50 = 5.3 nM T97719 COU73Y 71226944 IC50 = 13 nM T97719 C15FZU 71227026 IC50 = 377 nM T97719 CSB2N6 71235464 IC50 = 3.3 nM T97719 C40JOZ 71235465 IC50 = 14 nM T97719 C5YX9S 71450146 IC50 = 2 nM T97719 CQR24F 71453784 IC50 = 1050 nM T97719 C6LH8Q 71455522 IC50 = 5 nM T97719 CL9YX8 71455523 IC50 = 12 nM T97719 C7C5KR 71459146 IC50 = 15 nM T97719 CO0U6L 71473856 IC50 = 8 nM T97719 CMEH30 71473900 IC50 = 5 nM T97719 CVET45 71473952 IC50 = 23 nM T97719 CPV31M 71473953 IC50 = 44 nM T97719 CH8NC9 71473954 IC50 = 9.9 nM T97719 C2PMJ7 71474167 IC50 = 4 nM T97719 C9U1ZP 71474168 IC50 = 0.8 nM T97719 CZ20PT 71474283 IC50 = 5.9 nM T97719 C8S2WR 71474333 IC50 = 290 nM T97719 CGL3O6 71474335 IC50 = 0.6 nM T97719 C6C0ED 71526523 Ki = 0.32 nM T97719 C9ILH0 71526524 Ki = 0.43 nM T97719 CC3JG4 71526687 Ki = 0.37 nM T97719 C1NPL0 71552941 IC50 > 30000 nM T97719 CA4PS8 71552942 IC50 > 30000 nM T97719 C3UA9C 71553011 IC50 = 30000 nM T97719 CEZ15Y 71553012 IC50 = 25670 nM T97719 CVIA91 71553085 IC50 = 30000 nM T97719 C1TR3O 71553152 IC50 = 30000 nM T97719 C8I9RX 71554042 Ki = 0.65 nM T97719 CAYK39 71555872 IC50 = 39 nM T97719 C7ZR4F 71555873 IC50 = 14 nM T97719 C82JZR 71555942 IC50 = 18 nM T97719 CK5L4A 71555944 IC50 = 8563 nM T97719 C05AUY 71555945 IC50 = 25 nM T97719 CA60YZ 71556002 IC50 = 20 nM T97719 CUOQ40 71556003 IC50 = 4946 nM T97719 CNVU70 71556004 IC50 = 166 nM T97719 CP0BZ1 71556006 IC50 = 11 nM T97719 CMAE80 71556057 IC50 = 47 nM T97719 CG7XR2 71556058 IC50 = 47 nM T97719 C3VRD2 71556060 IC50 = 24 nM T97719 CT1AB4 71556116 IC50 = 233 nM T97719 CC0W9V 71556633 IC50 = 16 nM T97719 CLO1K4 71556702 IC50 = 36 nM T97719 C79ITZ 71556766 IC50 = 208 nM T97719 C3S0AK 71556770 IC50 = 22 nM T97719 C3SCM1 71556835 IC50 = 48 nM T97719 C4TS8W 71557106 Ki = 1.3 nM T97719 C0DXC9 71558702 Ki = 6.3 nM T97719 C6C8KF 71558854 Ki = 1.8 nM T97719 C1UJA7 71558855 Ki = 6.9 nM T97719 CA0JH1 71559158 Ki = 0.43 nM T97719 C1SR5V 71576693 Ki = 3.2 nM T97719 C0I8ZY 71721544 IC50 = 0.67 nM T97719 C5O3GQ 71731698 IC50 = 6.4 nM T97719 CW0U1X 71731701 IC50 = 2.2 nM T97719 CS27TG 71731982 IC50 = 43 nM T97719 C4X1CP 71748056 Ki = 14.2 nM T97719 C1T5AI 71760912 IC50 = 1 nM T97719 CF04BD 71765399 IC50 = 850000 nM T97719 CZM1K4 71765510 IC50 = 5.6 nM T97719 C4KV0T 71765585 EC50 = 92 nM T97719 C5MJ0H 71765626 IC50 = 2 nM T97719 C6WU5A 71769203 IC50 = 5600 nM T97719 CKO8S6 71815907 IC50 = 13.5 nM T97719 CZU45Y 72165218 IC50 = 101 nM T97719 C5WYP9 72188715 IC50 = 8.3 nM T97719 C54XWG 72190869 IC50 = 3.1 nM T97719 CTA6P1 72191176 IC50 = 1.1 nM T97719 C46RQD 72191792 IC50 = 5.5 nM T97719 C0LAS6 72191795 IC50 = 1.2 nM T97719 C18RFO 72193307 IC50 = 6.8 nM T97719 CDWL69 72193608 IC50 = 21 nM T97719 C9TUP2 72201774 IC50 = 13 nM T97719 C9OQ2I 72710839 IC50 > 10000 nM T97719 CX75YR 73352604 IC50 = 316.23 nM T97719 CDNQ20 73388819 IC50 = 1.3 nM T97719 C0ZJV3 73389638 IC50 = 1.9 nM T97719 CVRQ65 73438218 IC50 = 6.6 nM T97719 CLQN18 73438269 IC50 = 1.08 nM T97719 CX87NM 73438270 IC50 = 3.76 nM T97719 CYML76 73438271 IC50 = 0.903 nM T97719 CE85VI 73438272 IC50 = 1.48 nM T97719 C2THR4 73438379 IC50 = 31.2 nM T97719 CF6QG1 73602845 IC50 = 7.15 nM T97719 CDN83F 73707530 Ki = 2 nM T97719 CX1LR9 73774633 IC50 = 0.25 nM T97719 CCQN01 73775788 IC50 = 25.3 nM T97719 CHF08G 73775789 IC50 = 79.1 nM T97719 COL37D 73775921 IC50 = 10.7 nM T97719 CVQW20 73775923 IC50 = 37.2 nM T97719 C5U4AF 73776059 IC50 = 16.3 nM T97719 CXW54V 73776061 IC50 = 16.4 nM T97719 CD83FL 73776204 IC50 = 38.6 nM T97719 CG84BR 73776205 IC50 = 17.4 nM T97719 C1P3DO 73776206 IC50 = 115 nM T97719 CN5D1R 73776207 IC50 = 6.01 nM T97719 CO1C8Y 73776208 IC50 = 12.3 nM T97719 CGC46K 73776360 IC50 = 24.5 nM T97719 CS9BQ1 74222426 IC50 = 21 nM T97719 CO0V6K 74222427 IC50 = 1.5 nM T97719 CBE71O 74222509 IC50 = 7.6 nM T97719 CM02PA 74222510 IC50 = 0.37 nM T97719 CWLT81 74222511 IC50 = 33 nM T97719 C4XSG8 74222512 IC50 = 0.41 nM T97719 CBT4M6 74222513 IC50 = 2.7 nM T97719 C53AFH 74222599 IC50 = 2.3 nM T97719 CDJ2U1 75203907 IC50 < 10 nM T97719 CBRK81 75204377 IC50 = 0.17 nM T97719 CF26RG 76901709 Ki = 1.2 nM T97719 CO3V8L 77844057 IC50 = 13 nM T97719 CY2I8Q 77844118 IC50 = 4.11 nM T97719 CRGK76 77844121 IC50 = 265 nM T97719 C4ISQ7 77844176 IC50 = 318 nM T97719 C1S9WZ 77844178 IC50 = 31 nM T97719 C0G9VL 77844179 IC50 = 222 nM T97719 C6DBN5 77844241 IC50 = 30.6 nM T97719 CN28TW 78318226 IC50 < 1 nM T97719 CCJ3P8 78318227 IC50 = 1.3 nM T97719 CQFR81 78318278 IC50 < 1 nM T97719 CBQ9L7 86276271 IC50 < 0.5 nM T97719 C3B1EZ 86280660 IC50 = 8 nM T97719 COD2E9 86294808 IC50 = 17000 nM T97719 C3OU4B 86302101 IC50 = 63 nM T97719 CPG3A5 86302574 IC50 > 30000 nM T97719 C1CBD9 86342498 IC50 = 20 nM T97719 C1M7NF 86342499 IC50 = 9 nM T97719 CE1VD9 86342500 IC50 = 28 nM T97719 CNZU96 86342680 IC50 = 37 nM T97719 CD2V1S 86342681 IC50 = 564 nM T97719 CT0BM6 86342682 IC50 = 124 nM T97719 CN43WE 86342683 IC50 = 472 nM T97719 C74DWF 86342866 IC50 = 254 nM T97719 CK1G0U 86567260 Ki = 1.8 nM T97719 CV0SZ5 86567261 Ki = 0.96 nM T97719 CI1QK2 86580532 IC50 = 1.2 nM T97719 CRA17V 86580533 IC50 = 0.27 nM T97719 CI30UB 86580691 IC50 = 1.5 nM T97719 CJ24PC 86580692 IC50 = 2.2 nM T97719 CN08AB 86580693 IC50 = 240 nM T97719 CZQR95 86582648 IC50 = 11 nM T97719 C50NMW 86582649 IC50 = 4 nM T97719 CR12AD 86699873 IC50 = 139 nM T97719 C3KJI6 86721755 IC50 = 9 nM T97719 CB7C6T 86721760 IC50 = 0.2 nM T97719 CJUZ46 86721780 IC50 = 160 nM T97719 CIJ5H0 86721782 IC50 > 100000 nM T97719 CPUW96 86721788 IC50 = 730 nM T97719 CW8I1N 86721789 IC50 = 18 nM T97719 CMK52I 86721807 IC50 = 2.1 nM T97719 C1IXU4 86721808 IC50 = 5.5 nM T97719 CN1KU6 86721813 IC50 = 1200 nM T97719 CZ5J3N 86721820 IC50 = 14 nM T97719 COA34E 86721822 IC50 = 9.9 nM T97719 CTYW83 86724331 IC50 < 10 nM T97719 CTY9E7 86762906 IC50 = 550 nM T97719 C02UGP 87056204 IC50 = 0.39 nM T97719 CR08QT 89266687 IC50 = 143 nM T97719 CV5XT9 89266735 IC50 = 1500 nM T97719 C98MTY 89266756 IC50 = 660 nM T97719 CHO8S0 89266780 IC50 = 1510 nM T97719 C39VWO 89266843 IC50 = 21 nM T97719 CN25CP 89285825 IC50 = 150 nM T97719 CSG38E 89455222 IC50 = 2.2 nM T97719 CT8I9U 89455387 IC50 = 23.9 nM T97719 C2LW7J 89548692 IC50 = 16.1 nM T97719 CW5YJ9 89548700 Ki = 0.8 nM T97719 C1HW4B 89735655 IC50 = 13000 nM T97719 C9MO1Y 89906279 IC50 < 10 nM T97719 C3YID4 89968957 IC50 = 3.2 nM T97719 CT18GX 89994856 IC50 = 1.9 nM T97719 CI5WT1 90001694 IC50 = 4 nM T97719 CTMO59 90008542 IC50 = 2.6 nM T97719 C3BL8D 90008602 IC50 = 6 nM T97719 C79KGU 90008606 IC50 = 5.1 nM T97719 C3T1UQ 90008615 IC50 = 11.7 nM T97719 CEF98J 90008863 IC50 = 5.4 nM T97719 C07CZK 90054287 IC50 = 1 nM T97719 CR3XL7 90119070 IC50 = 176 nM T97719 CLK3O0 90119255 IC50 = 170 nM T97719 CO2FV0 90119264 IC50 = 0.18 nM T97719 C3RL4C 90136268 IC50 = 61 nM T97719 C4ME0V 90136282 IC50 = 1.6 nM T97719 CY0T6O 90136348 IC50 = 3.7 nM T97719 CTPY64 90234618 IC50 = 101 nM T97719 CP4S1M 90244576 IC50 < 10 nM T97719 CJB9Q8 90283189 IC50 = 1.1 nM T97719 CD2VO4 90311700 IC50 = 294 nM T97719 CP0X1V 90311949 IC50 = 0.9 nM T97719 CJ27GT 90467690 IC50 = 2.3 nM T97719 CN7CG9 90644798 IC50 = 1106 nM T97719 CYAI75 90644799 IC50 = 2153 nM T97719 CLZ71J 90644800 IC50 = 133 nM T97719 C19HKY 90644801 IC50 = 304 nM T97719 C3MU1B 90644802 IC50 = 53 nM T97719 CI0VF7 90644803 IC50 = 52 nM T97719 COA7S0 90644804 IC50 = 8 nM T97719 CY5Z3V 90644805 IC50 = 15 nM T97719 CGIL57 90644806 IC50 = 14 nM T97719 CUDB61 90644807 IC50 = 1410 nM T97719 C4Q3ZA 90644808 IC50 = 45 nM T97719 CMZ01N 90644809 IC50 = 9 nM T97719 CXQ3V4 90644810 IC50 = 15 nM T97719 CA90YJ 90644811 IC50 = 15 nM T97719 CAH2N9 90644812 IC50 = 18 nM T97719 C7N6HP 90644813 IC50 = 11 nM T97719 CU03MC 90656042 IC50 = 67 nM T97719 CF0C1K 90656043 IC50 = 12700 nM T97719 CFQ97Y 90656044 IC50 = 150 nM T97719 C5M2LN 90656045 IC50 > 50000 nM T97719 CTAL51 90656046 IC50 > 50000 nM T97719 C5DV2G 90656047 IC50 = 38 nM T97719 CC5UO8 90656048 IC50 = 213 nM T97719 C1IA4Z 90656049 IC50 = 574 nM T97719 C3PJ2I 90656050 IC50 = 64 nM T97719 CQX17K 90656051 IC50 = 25 nM T97719 CY45AL 90656052 IC50 = 28 nM T97719 C39BDP 90656053 IC50 = 17 nM T97719 CDR9B1 90656054 IC50 = 143 nM T97719 CV6C8G 90656055 IC50 = 43 nM T97719 CX2P0H 90656056 IC50 = 87 nM T97719 CN1B9K 90656057 IC50 = 126 nM T97719 CZ5A9D 90656058 IC50 = 19 nM T97719 CL3MH1 90656059 IC50 = 170 nM T97719 CKO3R1 90656060 IC50 = 140 nM T97719 COI9D2 90656061 IC50 > 50000 nM T97719 CX3A5W 90656062 IC50 = 29000 nM T97719 CI9WR3 90656063 IC50 = 970 nM T97719 C2C6EQ 90656064 IC50 = 33 nM T97719 C8L4EH 90656065 IC50 = 65 nM T97719 C8UCD2 90656066 IC50 = 26 nM T97719 CP5E9X 90656067 IC50 = 32 nM T97719 CD4FM8 90656068 IC50 = 48 nM T97719 C9WO2A 90656069 IC50 = 83 nM T97719 CN9VX7 90656070 IC50 = 169 nM T97719 CZJB24 90656071 IC50 = 109 nM T97719 C9Y5CR 90656072 IC50 = 77 nM T97719 CPRI81 90656073 IC50 = 35 nM T97719 CM5F7W 90656074 IC50 = 18 nM T97719 C15HEM 90656075 IC50 = 49 nM T97719 CG9I7R 90656076 IC50 = 27 nM T97719 C4OB0T 90656077 IC50 = 41 nM T97719 CF89DA 90664659 IC50 = 15500 nM T97719 C90JVH 91799688 IC50 = 1.4 nM T97719 C6J0GR 91809511 EC50 = 28600 nM T97719 CED37U 91885524 IC50 = 15 nM T97719 C64SIO 92042864 IC50 = 794 nM T97719 C39PCS 101898032 IC50 = 4.8 nM T97719 CAKD54 102594000 IC50 = 75.6 nM T97719 C6TWN0 117668201 IC50 = 150 nM T97719 CM7C3W 117668218 IC50 = 17 nM T97719 CTK65N 117668270 IC50 = 8 nM T97719 C63LHQ 117668291 IC50 = 0.32 nM T97719 CP3VQ6 117668361 IC50 = 860 nM T97719 C0V3ZB 117676956 IC50 = 0.13 nM T97719 CO4Z3X 117676961 IC50 = 0.19 nM T97719 C7RUS2 117676973 IC50 = 0.15 nM T97719 CB4XM9 117676974 IC50 = 14 nM T97719 C3NI4J 117676976 IC50 = 0.36 nM T97719 C3AX9V 117676992 IC50 = 34 nM T97719 C5LWU4 117677006 IC50 = 0.8 nM T97719 CNOR97 117761007 IC50 = 2.6 nM T97719 CT8Y1R 117773317 IC50 = 1.1 nM T97719 CV69NM 117778362 IC50 < 0.3 nM T97719 C8Y5ZX 117778486 IC50 = 8.3 nM T97719 CIH2K3 117780573 IC50 = 2.5 nM T97719 C5B3CM 117781182 IC50 = 4.2 nM T97719 C30KSM 117781201 IC50 = 4.7 nM T97719 CT68XG 117785578 IC50 = 0.62 nM T97719 C7C6KO 117785630 IC50 = 4.3 nM T97719 C0EJ2H 117785631 IC50 = 4 nM T97719 CL91NV 117785647 IC50 = 1.6 nM T97719 C41YCU 117785685 IC50 = 3.8 nM T97719 C4K5WY 117785740 IC50 = 0.81 nM T97719 CSC8F7 117785816 IC50 = 34 nM T97719 CFZ0P3 117785848 IC50 = 15 nM T97719 CA0G4U 117787055 IC50 = 80 nM T97719 C2EKR6 117802839 IC50 = 2.1 nM T97719 C3FY8A 117838708 IC50 = 0.58 nM T97719 C7VDL3 117838709 IC50 = 0.53 nM T97719 C0BI1C 117838710 IC50 = 0.49 nM T97719 C73JCL 117838721 IC50 = 0.51 nM T97719 CT5L8Z 117925826 IC50 = 1.7 nM T97719 C8HYU9 117926195 IC50 = 2.6 nM T97719 C45OGJ 117926401 IC50 = 1.4 nM T97719 CPD57Q 117948653 IC50 = 0.4 nM T97719 CB4R8H 117948656 IC50 = 20.2 nM T97719 C34FKB 118025462 IC50 = 142 nM T97719 CUQS80 118025552 IC50 = 217 nM T97719 C1KGB4 118025559 IC50 = 584 nM T97719 CDF6L7 118025606 IC50 = 891 nM T97719 CGX1T6 118025676 IC50 = 7 nM T97719 C1IL8Q 118025680 IC50 = 86 nM T97719 C79ZBM 118025723 IC50 = 14 nM T97719 C6HO9P 118025760 IC50 = 67 nM T97719 CM4Z5V 118025790 IC50 = 1970 nM T97719 CX4W9A 118025823 IC50 = 104 nM T97719 C3FG4U 118025830 IC50 = 84 nM T97719 CM3JO2 118025835 IC50 = 123 nM T97719 CKR9G1 118025928 IC50 = 27 nM T97719 C5TQU3 118025943 IC50 = 12 nM T97719 C68YAU 118026010 IC50 = 43 nM T97719 CJ6ZB1 118038061 IC50 = 180 nM T97719 CQ0XS5 118038146 IC50 = 32 nM T97719 CZIS42 118038175 IC50 = 4.1 nM T97719 CZP8A2 118038240 IC50 = 0.09 nM T97719 CYC26N 118038298 IC50 = 4.4 nM T97719 C6O1JB 118038376 IC50 = 4.3 nM T97719 CFE6M2 118038416 IC50 = 0.8 nM T97719 C5HYV8 118038480 IC50 = 11 nM T97719 CC9W3M 118038535 IC50 = 25 nM T97719 C1RT3W 118038598 IC50 = 16.2 nM T97719 CXF0P7 118038619 IC50 = 1.9 nM T97719 CA3B9Z 118038785 IC50 = 500 nM T97719 CF8DV9 118039033 IC50 = 5900 nM T97719 C0D3QO 118039090 IC50 > 6000 nM T97719 CF31OY 118039156 IC50 = 430 nM T97719 C2WQ4G 118039220 IC50 = 2.3 nM T97719 CTU3K2 118043167 IC50 = 2.8 nM T97719 C32TIM 118043177 IC50 = 13 nM T97719 CMR1B0 118043198 IC50 = 1.3 nM T97719 CYQ54O 118043226 IC50 = 40 nM T97719 CPU7C0 118043263 IC50 = 1.9 nM T97719 CR2XJ5 118043265 IC50 = 1.3 nM T97719 CQ1L8G 118043278 IC50 = 10000 nM T97719 C4HQ5C 118043312 IC50 = 2.2 nM T97719 CB4A6H 118043313 IC50 = 1.6 nM T97719 CB40XP 118043323 IC50 = 0.5 nM T97719 CO0HE8 118107408 IC50 = 7.5 nM T97719 CE37KU 118107427 IC50 = 1.8 nM T97719 CJ1UV7 118107429 IC50 = 8.7 nM T97719 CTA7N8 118107436 IC50 = 0.9 nM T97719 C49LKY 118107459 IC50 = 5 nM T97719 C5VDB3 118107478 IC50 = 3.7 nM T97719 CR6ND3 118107479 IC50 = 32 nM T97719 CMX3U8 118107483 IC50 = 1.3 nM T97719 C0YW3E 118107484 IC50 = 86 nM T97719 CK9F4X 118107489 IC50 = 104 nM T97719 CYAD17 118107490 IC50 = 91 nM T97719 CJGT03 118346182 IC50 = 105 nM T97719 C02DGP 118346184 IC50 = 155 nM T97719 CU6NE2 118346192 IC50 = 19.1 nM T97719 CW25VP 118346194 IC50 = 17.7 nM T97719 CPJX70 118722806 IC50 = 1600 nM T97719 CPUT35 118722848 IC50 = 431 nM T97719 CA6KN9 118722849 IC50 = 1030 nM T97719 CT16GW 118722850 IC50 > 5000 nM T97719 CF59DR 118722851 IC50 = 818 nM T97719 CHD92M 118722852 IC50 = 171 nM T97719 COH06T 118722854 IC50 > 5000 nM T97719 C13XBH 118722855 IC50 > 5000 nM T97719 C48XIV 118727100 IC50 < 0.5 nM T97719 CM2HX1 118727101 IC50 = 0.5 nM T97719 C3F1AI 118728082 IC50 = 5.6 nM T97719 CVG7K0 118728083 IC50 = 3.2 nM T97719 C9V6TB 118728174 IC50 = 1568 nM T97719 C42HQG 118728175 IC50 = 79 nM T97719 COZ6D3 118728176 IC50 = 73.9 nM T97719 C8GAN5 118728177 IC50 = 58.3 nM T97719 CGR39I 118728178 IC50 = 135.5 nM T97719 C72MTN 118728179 IC50 = 41.7 nM T97719 CE39IR 118728180 IC50 = 15 nM T97719 CZUK91 118728340 IC50 = 4600 nM T97719 CF1I8Y 118728341 IC50 = 860 nM T97719 CXN4L5 118728342 IC50 = 225 nM T97719 CYIW78 118728343 IC50 = 40 nM T97719 CSDN72 118728344 IC50 = 30 nM T97719 CEZ9I1 118728345 IC50 = 90 nM T97719 CMF71L 118728346 IC50 = 150 nM T97719 CD1L2J 118728347 IC50 = 340 nM T97719 C7HNK8 118728348 IC50 = 190 nM T97719 CN4O3J 118728349 IC50 = 490 nM T97719 C25UBH 118728350 IC50 = 650 nM T97719 C6VLK2 118728351 IC50 = 43 nM T97719 CP8RC3 118728352 IC50 = 210 nM T97719 C3OIW8 118728353 IC50 = 54 nM T97719 CD3QC7 118728354 IC50 = 10 nM T97719 C2XI0G 118728355 IC50 = 60 nM T97719 CMY1F0 118728356 IC50 = 50 nM T97719 CO3EX8 118729088 IC50 = 4.3 nM T97719 CUX3Q5 118729089 IC50 = 7.8 nM T97719 C3HJC0 118729090 IC50 = 0.61 nM T97719 CGS36E 118729091 IC50 = 4.8 nM T97719 C13YHN 118729092 IC50 = 4700 nM T97719 CDKA65 118729174 IC50 = 10 nM T97719 C75QXY 118729175 IC50 = 50.8 nM T97719 C0JVF5 118729176 IC50 = 31.6 nM T97719 CR4WD5 118729177 IC50 = 12 nM T97719 CX0C5K 118729178 IC50 = 69 nM T97719 CTQ16U 118729179 IC50 = 118.8 nM T97719 CL7K5B 118729182 IC50 = 74 nM T97719 CR3A4I 118729183 IC50 = 1357 nM T97719 COR4G6 118729184 IC50 = 77.8 nM T97719 CWJ72S 118729185 IC50 = 46 nM T97719 C6D1WK 118729186 IC50 = 96.5 nM T97719 CGZ4S0 118729187 IC50 = 57.1 nM T97719 CS82YE 118729188 IC50 = 15.3 nM T97719 CF03VI 118729189 IC50 = 7 nM T97719 CYF9K8 118729190 IC50 = 25.2 nM T97719 CV42FJ 118729191 IC50 = 26 nM T97719 CFM07R 118729192 IC50 = 7.9 nM T97719 C47YUJ 118729193 IC50 = 11 nM T97719 COKJ09 118729194 IC50 = 69.7 nM T97719 CCWN20 118729195 IC50 = 574 nM T97719 C3X4GU 118729196 IC50 > 5000 nM T97719 CQCX41 118737057 IC50 = 67 nM T97719 CY8N5B 121293751 IC50 = 0.21 nM T97719 C12LTV 121293832 IC50 = 34 nM T97719 CX05DR 121293857 IC50 = 0.077 nM T97719 C37DUM 121293882 IC50 = 0.38 nM T97719 C86FHD 121293911 IC50 = 0.59 nM T97719 C9VM5J 121293927 IC50 = 81 nM T97719 C5VBP2 121293929 IC50 = 6 nM T97719 CU3Z6N 121293943 IC50 = 0.23 nM T97719 C1HKI5 121293949 IC50 = 0.11 nM T97719 CF7ZJ6 121293963 IC50 = 63 nM T97719 C0JQW1 121294046 IC50 = 1.2 nM T97719 CXQR89 121294143 IC50 = 0.14 nM T97719 CFS3E4 121294208 IC50 = 92 nM T97719 C4H3YT 121294217 IC50 = 12 nM T97719 C46DBJ 121362063 IC50 = 0.86 nM T97719 COGV39 121362167 IC50 = 0.39 nM T97719 CW4PG2 121362179 IC50 = 0.54 nM T97719 CO9SQ6 121454909 IC50 = 0.4 nM T97719 C63CXY 121454977 IC50 = 132 nM T97719 CH0X4Z 121454982 IC50 = 1 nM T97719 CD1S0Q 121455095 IC50 = 0.4 nM T97719 CNV26K 121455511 IC50 = 0.4 nM T97719 CYN8D9 121455521 IC50 = 0.1 nM T97719 CA59TF 121455523 IC50 = 0.2 nM T97719 C9ZTE0 121455568 IC50 = 1.3 nM T97719 C6XYK5 121455572 IC50 = 11 nM T97719 CBKR90 121455587 IC50 = 3 nM T97719 CT0KS4 121455652 IC50 = 0.2 nM T97719 CK78BX 121455673 IC50 = 26 nM T97719 C9OJ4T 121455700 IC50 = 0.3 nM T97719 C8XD1R 121455701 IC50 = 0.5 nM T97719 CW35TI 121455794 IC50 = 0.3 nM T97719 C6ZT2U 121455810 IC50 = 0.4 nM T97719 CT2JS5 121455892 IC50 = 0.2 nM T97719 C7CDN6 121468958 IC50 = 0.6 nM T97719 CG1SO6 121468959 IC50 = 0.4 nM T97719 C6YME4 121468960 IC50 = 3.4 nM T97719 C3XF0K 121468962 IC50 = 0.6 nM T97719 C1P9EV 121468963 IC50 = 0.2 nM T97719 C7OB1W 121468964 IC50 = 0.3 nM T97719 C0EFG1 121468967 IC50 = 2.5 nM T97719 CYO26S 121468970 IC50 = 0.6 nM T97719 CK03NG 121468972 IC50 = 309 nM T97719 CTFK25 121468974 IC50 = 13.9 nM T97719 CKZE17 121468976 IC50 = 62 nM T97719 CFM73S 121468978 IC50 = 0.8 nM T97719 CT2X7E 121481190 IC50 = 2.6 nM T97719 CZI09K 121499156 IC50 = 30 nM T97719 C7QE2J 121513893 IC50 = 421 nM T97719 CLPI09 122180346 EC50 > 50000 nM T97719 C6HKR2 122186249 IC50 > 10000 nM T97719 CL8UG5 122186250 IC50 > 10000 nM T97719 C0R5NS 122186251 IC50 > 10000 nM T97719 CC14AM 122186252 IC50 = 2295 nM T97719 CDUK97 122186253 IC50 > 10000 nM T97719 C6KWG4 122186254 IC50 > 10000 nM T97719 CHD5F2 122186255 IC50 = 1052 nM T97719 C9OWX5 122186256 IC50 = 107.4 nM T97719 CC41ON 122186257 IC50 = 176.2 nM T97719 C4P9NA 122186258 IC50 = 387.1 nM T97719 CD9E7X 122186259 IC50 = 699.2 nM T97719 CGQ1J9 122186260 IC50 = 279.7 nM T97719 C3J6BA 122186261 IC50 = 12.8 nM T97719 CKNF81 122186262 IC50 = 527.6 nM T97719 C7Y5EB 122186263 IC50 = 454.2 nM T97719 C7DW3G 122186264 IC50 = 291.5 nM T97719 C2SYA4 122186265 IC50 = 137 nM T97719 C84OGD 122186266 IC50 = 420.9 nM T97719 C4ZM7J 122186267 IC50 = 408.7 nM T97719 C8JT9S 122188509 IC50 = 12.2 nM T97719 CZN2V0 122188510 IC50 = 11.8 nM T97719 C7NJY1 122188511 IC50 = 9.5 nM T97719 C2LHC7 122188512 IC50 = 7.8 nM T97719 C5HY7G 122188513 IC50 = 7.4 nM T97719 CY5J4R 122188514 IC50 = 25.5 nM T97719 CLWJ56 122188515 IC50 = 54.9 nM T97719 CAJ19Q 122188516 IC50 = 21 nM T97719 CGRX10 122188517 IC50 = 9.9 nM T97719 C73RVY 122188518 IC50 = 1687 nM T97719 CH96TK 122188519 IC50 = 2867 nM T97719 CBS04E 122188520 IC50 = 3601 nM T97719 C0L9BY 122188628 IC50 = 455.7 nM T97719 C9P2HC 122188629 IC50 = 342.6 nM T97719 CNS5A6 122188630 IC50 > 10000 nM T97719 CJ27GC 122188631 IC50 = 2295 nM T97719 C1HUP9 122188632 IC50 = 1659 nM T97719 C8MBX1 122188633 IC50 = 853.9 nM T97719 C19LMB 122188634 IC50 = 183.3 nM T97719 CRB9U6 122188635 IC50 > 10000 nM T97719 C9M1ZH 122191198 IC50 = 16 nM T97719 CVWF79 122191199 IC50 = 28 nM T97719 CN0KS5 122191200 IC50 = 88 nM T97719 CD4RL5 122191223 IC50 = 39 nM T97719 CF2I6C 122191224 IC50 = 32 nM T97719 C4C9TS 122191225 IC50 = 30 nM T97719 C34CUW 122191226 IC50 = 55 nM T97719 CTC5D3 122191227 IC50 = 15 nM T97719 CDA73F 122191228 IC50 = 24 nM T97719 CS98FB 122191229 IC50 = 144 nM T97719 C02OZK 122191230 IC50 = 38 nM T97719 CU08AN 122191231 IC50 = 71 nM T97719 CO5T1L 122191232 IC50 = 59 nM T97719 C03BMP 122191233 IC50 = 103 nM T97719 CIS71B 122191234 IC50 = 44 nM T97719 CHR68P 122191235 IC50 = 127 nM T97719 C61RMU 122191236 IC50 = 101 nM T97719 C35WTN 122191237 IC50 = 13 nM T97719 CR5EC8 122191238 IC50 = 6.9 nM T97719 C1DN4E 122191239 IC50 = 32 nM T97719 C5J4PL 122191240 IC50 = 22 nM T97719 CFAY16 122191241 IC50 = 16 nM T97719 CLY87F 122191242 IC50 = 12 nM T97719 CN62UO 122191243 IC50 = 7.2 nM T97719 CH7P9T 122191634 IC50 = 3.8 nM T97719 CZY4G5 122191635 IC50 = 3.5 nM T97719 C6O2XI 122191636 IC50 = 9.4 nM T97719 CFKD32 122191637 IC50 = 3 nM T97719 CEY5J8 122191638 IC50 = 39 nM T97719 C4X7SD 122192466 IC50 > 10000 nM T97719 C0CGR8 122396707 IC50 = 6 nM T97719 C6JO4C 122474157 IC50 = 10.2 nM T97719 C0XB2E 122475292 IC50 = 15.1 nM T97719 C6QHB4 122484585 IC50 = 518 nM T97719 CRT93E 122484586 IC50 = 248 nM T97719 CF7ME6 122484587 IC50 = 982 nM T97719 CX8EC3 122484589 IC50 = 396 nM T97719 C2E8NC 122484594 IC50 = 145 nM T97719 CTX02B 122484677 IC50 = 996 nM T97719 CJ63LF 122484678 IC50 = 852 nM T97719 C6DP2N 122484680 IC50 = 6.2 nM T97719 C2SXK9 122484682 IC50 = 806 nM T97719 C8MJ4P 122484684 IC50 = 718 nM T97719 C1U2WJ 122484694 IC50 = 30 nM T97719 CJC73G 122484695 IC50 = 76 nM T97719 C4AUD3 122484700 IC50 = 359 nM T97719 CS58YZ 122484702 IC50 = 364 nM T97719 CX6KW7 122484733 IC50 = 349 nM T97719 CV63PN 122484734 IC50 = 0.8 nM T97719 C1NPL5 122484735 IC50 = 1.2 nM T97719 C01SPL 122484737 IC50 = 23 nM T97719 CME91S 122513214 IC50 = 0.7 nM T97719 C32TWI 122513222 IC50 = 12 nM T97719 CLM7K3 122604539 IC50 > 10000 nM T97719 C01JHI 122604566 IC50 > 10000 nM T97719 C6UY2L 122633880 IC50 > 10000 nM T97719 CC7P2W 122633900 IC50 = 437 nM T97719 C4E7VI 124176804 IC50 = 6.6 nM T97719 CGN3H7 127034237 IC50 = 5.65 nM T97719 CWQ5C6 127039627 IC50 = 6 nM T97719 CYXB27 127039628 IC50 = 6 nM T97719 CX8J3E 127043557 IC50 = 1070 nM T97719 C2OSC6 127044265 IC50 = 880 nM T97719 CW85CM 127044597 IC50 = 1320 nM T97719 C01ERK 127044779 IC50 = 70 nM T97719 C6H1GW 127045093 IC50 = 1800 nM T97719 CIU72D 127264586 IC50 = 24.5 nM T97719 CGQZ74 129048381 IC50 = 6873 nM T97719 C0XS4M 129896681 EC50 = 4.7 nM T97719 CGIT40 129896911 IC50 = 24 nM T97719 CFD38L 130247375 IC50 = 1000 nM T97719 CK8UP1 130247747 IC50 = 10 nM T97719 CJ01GR 130247785 IC50 <= 10 nM T97719 C9XE1Y 130247799 IC50 = 100 nM T97719 CART50 130248020 IC50 <= 10 nM T97719 CZYM59 130248042 IC50 <= 10 nM T97719 C3RP1U 130248888 IC50 >= 10000 nM T97719 C6NH7E 130271687 IC50 = 100 nM T97719 CXV7B5 130319034 IC50 = 89 nM T97719 C5LOI7 130362292 IC50 = 0.16 nM T97719 CB8X2L 130362298 IC50 = 59 nM T97719 CA46DB 130362493 IC50 = 0.46 nM T97719 C71KMN 130429150 IC50 = 1213 nM T97719 CSG8J3 130429224 IC50 = 334 nM T97719 C5PT1M 130429242 IC50 = 1380 nM T97719 C0UNO3 130429244 IC50 = 153 nM T97719 CGFK71 130429248 IC50 = 1.91 nM T97719 CEX8D1 130429250 IC50 = 526 nM T97719 C9J6ZK 130429255 IC50 = 271 nM T97719 C6OMB1 132204257 IC50 = 95 nM T97719 C36ZNH 132231744 IC50 = 1.1 nM T97719 C92EAB 132231777 IC50 = 0.079 nM T97719 C2WL6U 132231784 IC50 = 0.17 nM T97719 C87MJN 132231796 IC50 = 0.24 nM T97719 CT0ZP1 132231829 IC50 = 1.2 nM T97719 CQXU93 132231841 IC50 = 0.18 nM T97719 CV89JM 132231876 IC50 = 0.21 nM T97719 CU9P7O 132247592 IC50 = 4.5 nM T97719 CD6TW5 132550270 IC50 = 0.82 nM T97719 CRV07S 132597737 IC50 = 47.4 nM T97719 CGV9B8 134135637 IC50 = 112 nM T97719 C56UDO 134135820 IC50 > 100 nM T97719 CU7E8V 134136144 IC50 = 32.1 nM T97719 C9GWC2 134136895 IC50 = 10.6 nM T97719 CQ2B0H 134137093 IC50 = 11 nM T97719 C25WAP 134137307 IC50 = 0.4 nM T97719 CQ61HU 134137344 IC50 > 100 nM T97719 CX1DP2 134138676 IC50 = 1.23 nM T97719 CN1I6V 134140323 IC50 = 17.1 nM T97719 C0PN3R 134140590 IC50 = 19 nM T97719 CE43OI 134144225 IC50 = 0.5 nM T97719 C20RHY 134145268 IC50 = 2.6 nM T97719 C3KZV6 134146771 IC50 > 100 nM T97719 C0F7OT 134149340 IC50 = 410 nM T97719 C10LWI 134151050 IC50 > 100 nM T97719 C43FPY 134151089 IC50 = 0.5 nM T97719 C1C7PJ 134152686 IC50 = 63 nM T97719 CG8OY3 134153160 IC50 > 100 nM T97719 C5HMI8 134153342 IC50 = 21.6 nM T97719 CUD7A8 134155908 IC50 = 97.1 nM T97719 C8CXZ9 134156759 IC50 = 13.2 nM T97719 C59HOQ 134277578 IC50 = 4.4 nM T97719 C0PZ5R 134277599 IC50 = 2.59 nM T97719 C7PWJ2 134277617 IC50 = 0.33 nM T97719 CRA2H1 134277633 IC50 = 1.34 nM T97719 CXJ8I0 134277643 IC50 = 0.64 nM T97719 C02RIA 134277647 IC50 = 0.63 nM T97719 CGH42R 134277652 IC50 = 0.62 nM T97719 COA14U 134277654 IC50 = 0.46 nM T97719 CQK0B5 134277685 IC50 = 1.8 nM T97719 C6S8VC 134277696 IC50 = 0.53 nM T97719 C49PIO 134277748 IC50 = 0.95 nM T97719 CD7VK4 134277767 IC50 = 0.7 nM T97719 CZ5E6L 134277773 IC50 = 0.66 nM T97719 C2CFK7 134277780 IC50 = 2.11 nM T97719 C6E7LW 134277790 IC50 = 0.94 nM T97719 C6T7NW 134277796 IC50 = 0.41 nM T97719 CU8ZP5 134277800 IC50 = 1.09 nM T97719 CTR4K6 134277828 IC50 = 0.68 nM T97719 C3AVH9 134551003 IC50 = 3 nM T97719 C4H5TL 134551018 IC50 = 6.1 nM T97719 C4TVJ1 134551049 IC50 = 3.3 nM T97719 C6HZF3 134551056 IC50 = 5.3 nM T97719 CX2VZ9 134551058 IC50 = 2.8 nM T97719 CN75GU 134611727 EC50 = 13300 nM T97719 C54FXD 134957362 IC50 > 10000 nM T97719 CTJ48K 135524085 IC50 > 10000 nM T97719 CUT1W7 135524168 IC50 > 10000 nM T97719 CY4D8I 135566504 Ki = 636.5 nM T97719 CZFA70 135611366 IC50 = 456 nM T97719 CG3UZ1 135927974 Ki > 1000 nM T97719 CRK8E5 136391507 IC50 = 1.9 nM T97719 CF3W4I 136928070 IC50 = 1000 nM T97719 CR69AU 136928128 IC50 = 2.7 nM T97719 C03VDE 136928142 IC50 = 2 nM T97719 C2RB4H 136961397 IC50 = 38.8 nM T97719 CMS37R 136961398 IC50 = 21.3 nM T97719 CTAS87 136983688 IC50 = 0.58 nM T97719 C8M2DL 136983691 IC50 = 9.5 nM T97719 CMOH82 136983718 IC50 = 0.64 nM T97719 C1JSX0 136983721 IC50 = 4.2 nM T97719 CRE05Z 136983730 IC50 = 232.6 nM T97719 CMP62O 136983732 IC50 = 1.6 nM T97719 CB26DO 136983736 IC50 = 4.2 nM T97719 C9J5KZ 136983740 IC50 = 1.6 nM T97719 CN7W2C 136983741 IC50 = 1.9 nM T97719 CPM64E 136983746 IC50 = 1.3 nM T97719 CM2IO7 136983748 IC50 = 0.38 nM T97719 C0F7EY 136983756 IC50 = 41 nM T97719 CID2U4 136983757 IC50 = 200 nM T97719 C60HNV 136983761 IC50 = 3.5 nM T97719 C4EKW0 136983767 IC50 = 0.24 nM T97719 CY89MV 137071299 IC50 = 11 nM T97719 C5MZV6 137189918 IC50 = 10910 nM T97719 CMCD09 137189935 IC50 = 46510 nM T97719 CT8EV4 137226337 IC50 = 3180 nM T97719 CXC69T 137321158 IC50 = 862 nM T97719 C3Z4AT 137321159 IC50 > 10000 nM T97719 C81LGX 137349435 IC50 = 7.5 nM T97719 C0A9SP 137353877 IC50 > 10000 nM T97719 C8WQ3V 137354009 IC50 = 365 nM T97719 CX4UT6 137475232 IC50 = 86 nM T97719 CBN69K 137475234 IC50 = 667 nM T97719 CFXK71 137475248 IC50 = 1697 nM T97719 CS5L0F 137475249 IC50 = 34 nM T97719 CM6P8G 137475250 IC50 = 19 nM T97719 CXKD71 137475453 IC50 = 63 nM T97719 CNI4D8 137475454 EC50 > 100 nM T97719 C21HSQ 137475456 IC50 = 273 nM T97719 C6P5AL 137475459 IC50 = 282 nM T97719 C1KSZ6 137475463 IC50 = 5.8 nM T97719 CTA26W 137475470 IC50 = 41 nM T97719 CPY52K 137475474 IC50 = 21 nM T97719 CUG84N 137475477 IC50 = 2610 nM T97719 C2FT1L 137475480 Ki = 6 nM T97719 C4K2UA 137475509 IC50 = 57 nM T97719 CL87BX 137475510 IC50 = 1261 nM T97719 CB2TR5 137475511 IC50 = 32 nM T97719 C36CKU 137475515 IC50 = 596 nM T97719 CIR4W0 137475517 IC50 = 65 nM T97719 C8PJ7Z 137475518 IC50 = 197 nM T97719 CE1O2J 137475520 IC50 = 3187 nM T97719 CE4ZT1 137475623 IC50 = 3736 nM T97719 CKIX38 137475632 IC50 = 4996 nM T97719 CLB03V 137475634 IC50 = 210 nM T97719 C4RZ6J 137475648 IC50 = 114 nM T97719 C4RH2N 137475657 IC50 = 1426 nM T97719 CJ5D6T 137475692 IC50 = 127 nM T97719 CC8H2P 137475700 IC50 = 244 nM T97719 CW12VL 137475702 IC50 = 1191 nM T97719 C4GYH0 137475704 IC50 > 10000 nM T97719 CZP8B9 137475873 IC50 = 68 nM T97719 CRKA51 137475874 IC50 = 187 nM T97719 CZ6YO7 137475875 IC50 = 76 nM T97719 C6J7QN 137632048 IC50 = 2410 nM T97719 CH9WK1 137632228 EC50 = 1576 nM T97719 C6VN7C 137632252 IC50 > 100 nM T97719 C0S6PX 137632398 IC50 > 100 nM T97719 CM28ZT 137632791 IC50 = 1.18 nM T97719 C30SZG 137633174 IC50 = 6 nM T97719 CXT73R 137633588 IC50 = 132 nM T97719 CRLT63 137633687 IC50 = 4 nM T97719 CZOD53 137633880 IC50 = 0.25 nM T97719 CI1E8V 137634241 IC50 = 5020 nM T97719 C9QGJ0 137634325 IC50 > 10000 nM T97719 CCM5R7 137634499 Ki = 1.8 nM T97719 C86CNU 137634727 IC50 = 0.23 nM T97719 C3UGD5 137635118 IC50 = 68.3 nM T97719 C6LPM5 137635156 IC50 = 0.5 nM T97719 C5VQM1 137635526 IC50 = 231 nM T97719 CJKI16 137635532 Ki = 0.58 nM T97719 CR2K6M 137635680 IC50 = 9.14 nM T97719 CYM4L6 137635963 IC50 = 0.5 nM T97719 C7BJY5 137636807 IC50 = 0.59 nM T97719 C7IL4D 137637204 IC50 = 0.7 nM T97719 CU9YQ3 137637635 IC50 = 911 nM T97719 C39XGQ 137637902 IC50 = 38 nM T97719 CWZY04 137638548 Ki = 3.3 nM T97719 CH1Y2J 137639108 IC50 = 0.42 nM T97719 C3ABE0 137639720 IC50 = 0.2 nM T97719 C4VDL6 137640150 IC50 = 0.92 nM T97719 CJ28YI 137640151 IC50 = 350 nM T97719 C40XZN 137640550 IC50 = 21.3 nM T97719 CQOW35 137641160 IC50 > 100 nM T97719 C7FWD3 137641710 Ki = 0.45 nM T97719 CNL87M 137641918 IC50 = 85.4 nM T97719 CBJX42 137642666 IC50 = 5.9 nM T97719 CJVX98 137642896 IC50 = 18.1 nM T97719 C9XWS8 137643176 IC50 = 78.6 nM T97719 CEYA97 137643185 IC50 = 22.4 nM T97719 C4DRX1 137643187 IC50 = 5030 nM T97719 CW5V3F 137643326 IC50 = 1.4 nM T97719 C2ID4H 137643621 IC50 = 6.7 nM T97719 CF5DH3 137643910 IC50 > 5000 nM T97719 CQZ6N3 137644623 IC50 = 22.6 nM T97719 C4I8HP 137644728 Ki = 2.5 nM T97719 CFU7S2 137645034 Ki = 1.8 nM T97719 CVFR40 137645536 Ki = 1.8 nM T97719 C20MIC 137645538 IC50 = 7.12 nM T97719 C3GC8E 137646450 IC50 = 0.3 nM T97719 C3BP6L 137646652 IC50 = 110 nM T97719 CB6H7D 137646812 IC50 = 9.7 nM T97719 C4X7BG 137647868 IC50 = 0.3 nM T97719 CBYF68 137647965 IC50 = 9.5 nM T97719 CN8F6I 137648044 IC50 = 20 nM T97719 C96CMS 137648135 IC50 = 0.6 nM T97719 CO89DX 137649100 IC50 = 0.8 nM T97719 COLY80 137649218 IC50 = 0.1 nM T97719 C3FWY7 137649370 IC50 = 3.4 nM T97719 CAGB21 137649664 IC50 > 10000 nM T97719 C2QYK3 137649872 IC50 = 3 nM T97719 CYI4T1 137650386 IC50 = 2.83 nM T97719 C0D9MO 137651114 IC50 = 7.3 nM T97719 CH9W6N 137651389 Ki = 5.97 nM T97719 C7THC2 137652002 Ki = 4 nM T97719 CINE03 137652514 IC50 = 26 nM T97719 CBS5J3 137652658 IC50 = 27.2 nM T97719 C28QUP 137652864 IC50 = 88.6 nM T97719 C62JYT 137653234 IC50 = 91.3 nM T97719 C7R1WL 137653505 IC50 = 27.3 nM T97719 C6YAM7 137653900 IC50 = 69 nM T97719 C9T8NA 137654497 IC50 = 12.1 nM T97719 C1SWN5 137654673 IC50 = 1.05 nM T97719 C8BDX5 137655281 IC50 = 0.4 nM T97719 CU7I4L 137655908 IC50 = 48.6 nM T97719 COH9N2 137656066 Ki = 1 nM T97719 C6UW8I 137656158 IC50 = 5 nM T97719 C3YLU8 137656342 IC50 = 2946 nM T97719 CGW9I0 137656387 IC50 = 5000 nM T97719 C1T7DU 137656692 IC50 = 10.4 nM T97719 C3N4YM 137656842 IC50 = 213 nM T97719 CR6J9O 137656849 IC50 = 1.2 nM T97719 C7YHC0 137657046 IC50 = 58.5 nM T97719 CW1J7N 137657095 IC50 = 1.2 nM T97719 CF9Q8V 137657300 IC50 = 12.1 nM T97719 CV13JT 137657722 IC50 = 7.1 nM T97719 CJH0B6 137658413 Ki = 4.2 nM T97719 C03AHL 137658850 IC50 = 0.3 nM T97719 C0GC8I 137658926 IC50 > 10000 nM T97719 CRA21G 137658982 IC50 > 10000 nM T97719 CUP8I0 137659174 IC50 = 11 nM T97719 C2ZB5H 137660502 IC50 = 4.94 nM T97719 C40WUE 137660864 Ki = 1 nM T97719 C29HIS 137661280 IC50 = 28.3 nM T97719 CJ0SU5 137661571 IC50 = 23.8 nM T97719 CSTV07 137662233 IC50 = 92.7 nM T97719 CU2L5H 138108525 EC50 > 10000 nM T97719 CB8FE3 138393376 IC50 = 1 nM T97719 CN0X5D 138454787 IC50 = 161 nM T97719 CUXO19 138617501 IC50 > 1000 nM T97719 CRWA29 139030520 EC50 = 42.7 nM T97719 C72TXN 139465220 IC50 <= 10 nM T97719 CBI6F5 139465310 IC50 = 10 nM T97719 C47UIT 139473914 IC50 <= 10 nM T97719 C3JYA8 139474172 IC50 <= 10 nM T97719 C3JWI7 139507347 IC50 = 2.8 nM T97719 C1N5QZ 141366015 IC50 = 7 nM T97719 C9ZYG8 141366083 IC50 = 9.3 nM T97719 COW01B 141366090 IC50 = 2 nM T97719 CH5NU8 141366112 IC50 = 5 nM T97719 C5E3OG 141366257 IC50 = 16 nM T97719 C7RME6 141366266 IC50 = 3 nM T97719 C65RGZ 141366278 IC50 = 5 nM T97719 CIQ96U 141478757 IC50 = 1300 nM T97719 CLY5A8 141496674 IC50 = 209.2 nM T97719 C1OTX5 141496811 IC50 = 102.4 nM T97719 CZS03J 141509623 IC50 = 136 nM T97719 C32ADR 141509628 IC50 = 119 nM T97719 CHV69N 141509629 IC50 = 80 nM T97719 CS7F1P 141509631 IC50 = 183 nM T97719 CX12GN 141509638 IC50 = 106 nM T97719 CVG92Q 141509639 IC50 = 200 nM T97719 CV8MJ3 141509640 IC50 = 50 nM T97719 CU51PI 141531440 IC50 = 203.1 nM T97719 C81RPA 141531442 IC50 = 481.2 nM T97719 CAT46B 141531443 IC50 = 180.3 nM T97719 CSU0P6 141622000 IC50 = 5 nM T97719 CCX7L5 141622014 IC50 = 5 nM T97719 CF1R6Z 141725864 IC50 = 12.8 nM T97719 C6UA7H 142357225 IC50 = 2.1 nM T97719 CMHX97 145331319 IC50 = 1.9 nM T97719 CVID46 145331320 IC50 = 31.9 nM T97719 CW1P9K 145331325 IC50 = 17.2 nM T97719 CDB9Y1 145331327 IC50 = 5.4 nM T97719 CG6V5Q 145331334 IC50 = 20.8 nM T97719 CGPH07 145331338 IC50 = 236.6 nM T97719 C6C5DF 145331339 IC50 = 21.8 nM T97719 CXCO76 145331341 IC50 = 2.4 nM T97719 CFY21D 145961655 EC50 = 5790 nM T97719 CQ86LZ 145963345 EC50 > 10000 nM T97719 CJ38PD 145964020 IC50 = 417.4 nM T97719 CE9ML8 145964464 IC50 = 3.1 nM T97719 CPU95I 145964675 IC50 = 0.6 nM T97719 COXI60 145966049 IC50 = 8800 nM T97719 CO7Y6G 145966466 IC50 = 40 nM T97719 CZJ6K7 145966487 IC50 = 100 nM T97719 CA5T8S 145966795 IC50 = 52 nM T97719 CTJE41 145966905 IC50 = 6.1 nM T97719 C4OD9Q 145967187 IC50 = 0.4 nM T97719 C8C9KB 145967601 IC50 = 18.11 nM T97719 CAIB20 145967604 IC50 = 49.23 nM T97719 CS6G9N 145967737 IC50 = 15.9 nM T97719 CEK76M 145967834 IC50 = 11.3 nM T97719 CIR2O4 145968647 IC50 = 20.85 nM T97719 CI0XK9 145968683 IC50 = 0.5 nM T97719 CZT26F 145969236 IC50 = 10.95 nM T97719 C1U0NB 145969251 IC50 = 7.95 nM T97719 C4QH6O 145969743 IC50 = 26.89 nM T97719 CBDL98 145969762 IC50 = 18.1 nM T97719 CZ9I5X 145969766 IC50 = 9.84 nM T97719 CJR62Q 145970555 IC50 = 22.18 nM T97719 CF12YE 145970801 IC50 = 89.62 nM T97719 CN76WO 145970945 IC50 = 45.35 nM T97719 C0BGW8 145971022 IC50 = 725.2 nM T97719 C9T8HZ 145971801 IC50 = 0.4 nM T97719 C8NCR2 145971905 IC50 = 2.2 nM T97719 CB5HF9 145972552 IC50 = 23.8 nM T97719 C50WPS 145972838 IC50 = 40.1 nM T97719 CJB41K 145973790 IC50 = 7300 nM T97719 CA7X9N 145973949 IC50 = 22 nM T97719 CP2EY5 145974012 IC50 = 62.6 nM T97719 C8XAG3 145974040 IC50 = 3.7 nM T97719 CS6WP7 145974982 IC50 = 0.41 nM T97719 C1E0IL 145975398 IC50 = 440 nM T97719 C4M6OX 145976007 IC50 = 0.8 nM T97719 CM3D2W 145976100 IC50 > 1000 nM T97719 CU1OX3 145976315 IC50 = 23.6 nM T97719 C5WJ0D 145976790 IC50 = 4.3 nM T97719 CI8WD9 145977263 IC50 = 3.5 nM T97719 C3ISA8 145977288 IC50 = 4.3 nM T97719 C8S7YH 145977937 IC50 = 50.4 nM T97719 CIV26F 145978013 IC50 = 7.4 nM T97719 C4Z3BX 145978513 IC50 = 0.4 nM T97719 CXE8H0 145979687 IC50 = 17.1 nM T97719 CE31VG 145979714 IC50 > 10000 nM T97719 C5WH9O 145979909 IC50 = 0.52 nM T97719 CA2CD1 145980524 IC50 = 89.32 nM T97719 CR43KU 145980943 IC50 = 10.5 nM T97719 CNDI08 145981275 IC50 = 0.6 nM T97719 C4O7LK 145982512 IC50 = 0.82 nM T97719 CL3R7U 145982901 IC50 = 217 nM T97719 C34LTV 145982927 IC50 = 0.1 nM T97719 C5VF8P 145983087 IC50 = 126.4 nM T97719 C35FMR 145983116 IC50 = 8.7 nM T97719 C0YFS6 145983170 IC50 = 11.2 nM T97719 C48ZXP 145983545 IC50 = 8.7 nM T97719 C8O1AM 145983591 IC50 = 153 nM T97719 CA20KM 145983867 IC50 = 159 nM T97719 CN7W3R 145984041 IC50 = 9.1 nM T97719 CM8Z7V 145984082 IC50 = 6.5 nM T97719 CN4H3U 145984330 IC50 = 3.5 nM T97719 CVCP14 145984386 IC50 = 1.1 nM T97719 C52FGO 145984982 IC50 = 12 nM T97719 CG4U3I 145985120 IC50 = 420.4 nM T97719 C7EV2P 145985201 IC50 = 36 nM T97719 CXQ2O9 145985661 IC50 = 90 nM T97719 CT6P1E 145986054 IC50 = 2.4 nM T97719 CID7Y4 145986342 IC50 = 39.8 nM T97719 C3TH4Z 145986350 IC50 = 38.17 nM T97719 C17TBU 145986946 IC50 = 31.3 nM T97719 C52AOJ 145987765 IC50 = 1 nM T97719 CG9AH0 145987953 IC50 = 23.2 nM T97719 CM1K2H 145988251 IC50 = 8 nM T97719 C9BX4U 145988956 IC50 > 10000 nM T97719 CNI4C6 145989069 IC50 = 1600 nM T97719 CL1IV0 145989334 IC50 = 0.6 nM T97719 CGB2F6 145989547 IC50 = 0.7 nM T97719 C82FRH 145989705 IC50 = 0.8 nM T97719 CLM9U8 145989960 IC50 > 100 nM T97719 CQH40O 145990342 IC50 = 0.7 nM T97719 CMP97L 145990518 IC50 < 0.5 nM T97719 C6LSR8 145990895 IC50 = 0.8 nM T97719 C8T5QK 145991122 IC50 = 16 nM T97719 C8EAO1 145991760 IC50 = 1.6 nM T97719 C71HFI 145992300 IC50 = 81.7 nM T97719 CYZ72C 145994233 IC50 = 0.5 nM T97719 C3U4FY 155510736 IC50 = 5.68 nM T97719 C3EK1O 155510821 IC50 = 263.7 nM T97719 CMT02R 155511053 IC50 = 30.7 nM T97719 CS2U6K 155511219 IC50 = 18.5 nM T97719 CF27EG 155511610 IC50 = 287 nM T97719 CLAN63 155511649 IC50 = 23.7 nM T97719 CH3N4R 155512268 IC50 = 63.2 nM T97719 C3TAO2 155512304 IC50 = 2.39 nM T97719 C0AN1O 155512752 IC50 = 880 nM T97719 CB0N3M 155513186 IC50 = 56.9 nM T97719 C2MD1Q 155513187 IC50 > 10000 nM T97719 CA7O4B 155513491 IC50 = 8 nM T97719 C7MYO1 155514069 IC50 = 11.1 nM T97719 CZK4R0 155514194 IC50 = 35.6 nM T97719 CMR01Y 155514274 IC50 = 8.9 nM T97719 C7AMX8 155514903 IC50 = 942 nM T97719 CJ2XU8 155515191 IC50 = 11 nM T97719 C9PK2F 155515251 IC50 = 2229 nM T97719 CAR70X 155516363 IC50 = 36.6 nM T97719 CPM06N 155516429 IC50 = 35.4 nM T97719 CI23DH 155516489 IC50 = 996 nM T97719 C0GA2M 155516495 IC50 = 72.8 nM T97719 C5PHO9 155516709 IC50 = 154.5 nM T97719 CWXG94 155517099 IC50 = 8300 nM T97719 CLT70D 155517651 IC50 = 9.7 nM T97719 C8V9IM 155517893 IC50 = 68.3 nM T97719 CNBF94 155518187 IC50 = 7300 nM T97719 C4SVP7 155518257 IC50 = 38109 nM T97719 C6PT7H 155518445 IC50 = 13.2 nM T97719 C6Z8AT 155518957 IC50 = 130.6 nM T97719 C3NA2I 155519537 IC50 = 3 nM T97719 CL67JW 155520152 IC50 = 11.6 nM T97719 CGP0T7 155520658 IC50 = 16.5 nM T97719 C9TU2A 155520832 IC50 = 9.67 nM T97719 CI7HF6 155520873 IC50 > 500 nM T97719 C8HMN5 155521132 IC50 = 1.8 nM T97719 CC6O8T 155521339 IC50 = 2422 nM T97719 CD6BW4 155521972 IC50 = 258 nM T97719 C3MB7J 155522852 IC50 = 80.3 nM T97719 CLYQ13 155523828 IC50 = 125.2 nM T97719 CCF73Y 155524267 IC50 = 206 nM T97719 CFZ71B 155524499 IC50 = 15 nM T97719 CM09ZA 155524938 IC50 = 150 nM T97719 C9HBS1 155525156 IC50 = 45.5 nM T97719 C1TXJ8 155525159 IC50 = 159 nM T97719 C4O6HM 155525406 IC50 = 122.6 nM T97719 C1W5PI 155525516 IC50 = 6754 nM T97719 CRT67D 155526236 IC50 = 26 nM T97719 CE3OH1 155527121 IC50 = 35 nM T97719 CXOC93 155527452 IC50 = 18.4 nM T97719 CE2T0A 155527963 IC50 = 862 nM T97719 CIOL97 155528057 IC50 = 637 nM T97719 CZ1NG6 155528141 IC50 = 115.2 nM T97719 CG64WY 155528210 IC50 = 51 nM T97719 C5TY7L 155528304 IC50 = 2000 nM T97719 CCL2W7 155528484 IC50 = 1.15 nM T97719 CK5JY6 155528755 IC50 = 29.9 nM T97719 CTM92N 155528887 IC50 = 68000 nM T97719 CL38EX 155529541 IC50 = 2.3 nM T97719 CUXA18 155529935 IC50 = 1481 nM T97719 CM3Z8Q 155530172 IC50 = 3.6 nM T97719 CL0US4 155530459 IC50 = 3.9 nM T97719 C2WCU6 155530774 IC50 = 1456 nM T97719 C8WQY6 155531004 IC50 = 7.36 nM T97719 CQD8I0 155531565 IC50 = 8.49 nM T97719 CB1R7F 155531721 IC50 = 0.2 nM T97719 CMV9N8 155533061 IC50 = 1290 nM T97719 C0JNV2 155533438 IC50 = 27.1 nM T97719 C1NGV5 155534208 IC50 = 270 nM T97719 CM0U3I 155534552 IC50 > 1000 nM T97719 C1K8RJ 155534556 IC50 = 2.5 nM T97719 CZ81CR 155534707 IC50 = 8529 nM T97719 CS4A8R 155535551 IC50 = 213 nM T97719 C5TYF1 155535789 IC50 > 500 nM T97719 C78MZC 155536330 IC50 = 2 nM T97719 CD0R7C 155536414 IC50 = 98.2 nM T97719 CJ1IR4 155536431 IC50 = 8.21 nM T97719 C3LC9I 155536820 IC50 = 1584.89 nM T97719 CAQB79 155537002 IC50 = 11000 nM T97719 C2CG1A 155537016 IC50 > 10000 nM T97719 C06LXE 155538200 IC50 = 62845 nM T97719 CCN3M1 155538205 IC50 = 1.44 nM T97719 CNC60O 155538282 IC50 = 240.8 nM T97719 C3V4LG 155538413 IC50 = 237 nM T97719 C0U5YH 155538856 IC50 = 23 nM T97719 CBI81T 155539300 IC50 > 500 nM T97719 CW9J0A 155539317 IC50 = 14.8 nM T97719 CW6G3P 155540991 IC50 = 13.9 nM T97719 CFL16S 155541157 IC50 = 19000 nM T97719 CH10DU 155542091 IC50 = 1469 nM T97719 CZJ89B 155542162 IC50 = 4.2 nM T97719 CJXD07 155542870 IC50 = 10.8 nM T97719 C3FI9X 155543272 IC50 = 5254 nM T97719 CW73EO 155543439 IC50 = 36 nM T97719 C7K0OW 155544589 IC50 = 1120 nM T97719 CK6OS8 155545032 IC50 = 4195 nM T97719 C6F4JP 155546501 IC50 = 28.3 nM T97719 CDN60A 155547934 IC50 > 500 nM T97719 C1HPS7 155548524 IC50 = 21045 nM T97719 C4U9BD 155548652 IC50 = 73 nM T97719 CX9M1U 155548660 IC50 = 83.6 nM T97719 C4DC0V 155548954 IC50 = 733 nM T97719 C2Z4SX 155549111 IC50 = 23.3 nM T97719 C9Z7AM 155549842 IC50 = 91.7 nM T97719 CU94IA 155550455 IC50 = 125 nM T97719 C9VL3E 155550614 IC50 = 37114 nM T97719 CM9F6A 155551058 IC50 = 11.1 nM T97719 CFC2U1 155551386 IC50 = 90 nM T97719 CG7PR3 155552009 IC50 = 283.5 nM T97719 CE9UZ4 155552131 IC50 = 16000 nM T97719 CH0OY2 155552417 IC50 = 1.9 nM T97719 C6LEU2 155552459 IC50 = 4100 nM T97719 CHNU54 155552592 IC50 = 134 nM T97719 C0HUL3 155552710 IC50 = 434 nM T97719 C8TK4O 155552924 IC50 = 31.1 nM T97719 CPR9B5 155553418 IC50 = 2671 nM T97719 C8RFE7 155553522 IC50 = 18.8 nM T97719 CE0GX5 155554136 IC50 = 5169 nM T97719 C87XLB 155554564 IC50 = 105 nM T97719 CCK0F7 155554945 IC50 = 48.6 nM T97719 CX41VR 155556272 IC50 = 150 nM T97719 CM7Q3F 155556300 IC50 = 0.536 nM T97719 CHF87X 155557221 IC50 = 19155 nM T97719 C0FE4G 155557988 IC50 = 74 nM T97719 C21GNS 155558056 IC50 = 3.8 nM T97719 CHBD73 155558571 IC50 = 89.4 nM T97719 CZK10J 155558893 IC50 = 2096 nM T97719 CPAV79 155559005 IC50 > 3000 nM T97719 C9KX4D 155559215 IC50 = 550 nM T97719 C4L6HQ 155559509 IC50 > 10000 nM T97719 C51IBQ 155560019 IC50 = 1607 nM T97719 CY7FH8 155560115 IC50 = 614 nM T97719 C3HF6R 155561374 IC50 = 12000 nM T97719 CHT92X 155562269 IC50 = 7.8 nM T97719 C0OA5R 155562881 IC50 = 41.9 nM T97719 CW4LI7 155563694 IC50 = 27822 nM T97719 CW56DX 155563904 IC50 = 385.9 nM T97719 CAC85T 155564156 IC50 > 10000 nM T97719 C71ILK 155565394 IC50 = 617 nM T97719 C26URQ 155566212 IC50 = 45 nM T97719 CD0EK2 155566233 IC50 = 6.9 nM T97719 CPAY80 155566268 IC50 = 161 nM T97719 C9S8JX 155566610 IC50 = 333 nM T97719 CB8PM4 155567091 IC50 = 21888 nM T97719 C49EVT 155567502 IC50 > 500 nM T97719 CU0VN4 155567699 IC50 = 1437 nM T97719 CDW02C 155567865 IC50 = 8.58 nM T97719 CBE0S8 155568469 IC50 > 500 nM T97719 CGU74Q 155569301 IC50 = 286 nM T97719 C1ZE2Y 155569446 IC50 = 5323 nM T97719 CBP05X 155569566 IC50 = 0.9 nM T97719 D01RHR 71519693 IC50 = 5 nM T97719 D01VFR 4708 IC50 = 5830 nM T97719 D04PEI 11467730 IC50 = 4100 nM T97719 D06BJG 71556703 IC50 < 4.4 nM T97719 D07OXC 11650194 IC50 = 19 nM T97719 D0E7VO 59627005 IC50 = 3.5 nM T97719 D0GN5Z 5281295 IC50 = 6020 nM T97719 D0H3JH 24857323 IC50 = 0.61 nM T97719 D0N0LN 46908026 IC50 = 13 nM T97719 D0O6OH 71553154 IC50 = 950 nM T97719 D0OZ2S 11785878 IC50 = 410 nM T06046 D08ZEB 2733 IC50 = 8700 nM T06046 D05QJT 9797017 IC50 = 466000 nM T06046 D07WGN 656912 Ki = 110 nM T06046 D0D3AI 39836 IC50 = 1500 nM T06046 D0V0NL 2146 IC50 = 72000 nM T06046 D0R5XK 9815538 Ki = 18.62 nM T06046 D0Y7VJ 2733506 IC50 = 2600 nM T06046 CHM9K2 4366 IC50 = 330 nM T06046 C9OF8C 5142 IC50 = 7000 nM T06046 C20EWK 15347 IC50 = 1200 nM T06046 CL81BQ 15348 IC50 = 3100 nM T06046 C6WDC5 15765 IC50 = 820 nM T06046 C5TXR9 27842 IC50 = 14700 nM T06046 C9NY7L 73046 IC50 = 650 nM T06046 C8CQW2 73742 IC50 = 1400 nM T06046 C7AB0Y 107968 IC50 = 400 nM T06046 CZXU91 118425 IC50 = 230 nM T06046 CP49UZ 132862 IC50 = 300 nM T06046 CT7M5K 135193 IC50 = 680 nM T06046 CWG0F1 152144 IC50 = 18900 nM T06046 CW72NB 203391 Ki = 11000 nM T06046 CG96BR 211124 IC50 > 50000 nM T06046 C23ABJ 262484 IC50 = 2800 nM T06046 C8B7YF 287208 IC50 > 50000 nM T06046 CC1X3J 317495 IC50 = 81 nM T06046 C3ZA0H 322632 IC50 = 10600 nM T06046 CV7K2N 322634 IC50 > 50000 nM T06046 C35JRN 449021 IC50 = 3500 nM T06046 C40ZOB 544920 IC50 > 50000 nM T06046 C9ABD3 656910 Ki = 107 nM T06046 CF7Z2I 656911 Ki = 80 nM T06046 C8SFX0 708870 IC50 > 50000 nM T06046 C39PAJ 764995 IC50 = 180 nM T06046 CNM06C 1375038 EC50 > 100000 nM T06046 C6U5SR 2733505 IC50 = 138000 nM T06046 C2B8KV 2778315 IC50 = 72400 nM T06046 C59BGS 2818222 Ki = 2600 nM T06046 CH5QU8 3016310 IC50 = 3600 nM T06046 C5L7GD 3636377 Ki = 38000 nM T06046 C4VNF7 3792909 IC50 = 30000 nM T06046 CUI4F5 4247236 IC50 = 300 nM T06046 C97INL 4262401 Ki > 50000 nM T06046 C6KW9G 4469991 IC50 = 5460 nM T06046 CLP5G9 8775318 Ki = 900 nM T06046 CI6O2G 8775930 Ki = 2700 nM T06046 C5GNH3 8776467 Ki = 1600 nM T06046 C5ATV1 9793824 IC50 = 2000 nM T06046 CC52JU 9794039 IC50 = 1900 nM T06046 C5Y0ZU 9795129 IC50 = 9000 nM T06046 CE62HS 9796600 IC50 = 5785 nM T06046 C4H6JA 9797393 IC50 = 5750 nM T06046 C3AWZ7 9815642 IC50 = 81000 nM T06046 C96UVG 9815901 Ki = 46000 nM T06046 CN6XG0 9816945 Ki = 4000 nM T06046 CQCA72 9818336 IC50 = 3710 nM T06046 CCS6E5 9819003 IC50 = 56660 nM T06046 CX7E2G 9823715 IC50 > 1000000 nM T06046 CHIO18 9834486 IC50 = 17200 nM T06046 CBZ95E 9837386 IC50 = 6200 nM T06046 CQF37H 9839201 IC50 = 1572 nM T06046 CP2IL5 9842658 Ki = 350 nM T06046 C80IET 9843967 IC50 = 887 nM T06046 CZMF39 9873870 IC50 = 80000 nM T06046 CAM64J 9881505 IC50 > 100000 nM T06046 C0JHT5 9905692 IC50 = 3713 nM T06046 CEF5Q9 9907534 IC50 = 31710 nM T06046 CR49WY 9920741 IC50 = 3300 nM T06046 CBA1D9 9927237 IC50 = 19000 nM T06046 C1LGZ2 9930200 IC50 = 49 nM T06046 C3PH5S 9931834 IC50 = 343400 nM T06046 C72OQJ 9942188 IC50 = 200 nM T06046 CGU01Y 9950094 IC50 = 36000 nM T06046 C1YG4Z 9990159 IC50 = 50 nM T06046 CNB2L4 9991061 Ki = 1600 nM T06046 CRD49Q 9991876 IC50 = 44000 nM T06046 C0Z2GX 10011896 IC50 = 1260 nM T06046 C74TYX 10013642 IC50 = 920 nM T06046 CL3Y5Z 10020993 IC50 = 6700 nM T06046 CYZJ64 10034809 IC50 = 870 nM T06046 C7YM4U 10060017 Ki = 270 nM T06046 CS7I1H 10068818 IC50 = 1500 nM T06046 C58LCS 10103217 IC50 > 50000 nM T06046 C0DW3A 10103242 IC50 = 2100 nM T06046 C3GVU2 10104005 IC50 = 9500 nM T06046 C9Z1HS 10149857 IC50 = 18197.01 nM T06046 CHT12V 10171540 IC50 = 45708.82 nM T06046 CD5NH1 10172593 IC50 = 66069.34 nM T06046 CJ97GV 10176386 Ki = 1100 nM T06046 C7NV2T 10192988 IC50 = 100000 nM T06046 CHJN87 10214800 IC50 = 8833 nM T06046 CHF49M 10215218 IC50 = 204173.79 nM T06046 CK7GN4 10219896 IC50 = 182000 nM T06046 CA68IC 10220131 IC50 = 57500 nM T06046 C1FZR9 10220855 IC50 = 79000 nM T06046 C3NPV0 10221335 IC50 = 7400 nM T06046 CAEK83 10248425 IC50 = 9400 nM T06046 C8P7WJ 10263292 IC50 = 34000 nM T06046 CBP8Q2 10265375 IC50 = 2300 nM T06046 CVTQ48 10286162 IC50 > 100000 nM T06046 CN42PW 10308710 IC50 = 87096.36 nM T06046 CS8T6Z 10313224 IC50 = 360 nM T06046 CJ3W7S 10330523 IC50 = 8420000 nM T06046 C31AYP 10330543 IC50 = 5800 nM T06046 CNKY10 10330544 IC50 = 2700 nM T06046 CWDA37 10358114 IC50 = 3533 nM T06046 C41RXN 10376219 IC50 = 19700 nM T06046 CALW76 10398017 IC50 = 578000 nM T06046 CIHA04 10398629 Ki = 250 nM T06046 C4P8EC 10400619 IC50 = 17000 nM T06046 CR47JC 10411355 IC50 = 6000 nM T06046 CK7FE5 10445220 IC50 = 160 nM T06046 C7E2VQ 10452321 IC50 = 900 nM T06046 CG94NE 10488346 IC50 = 47000 nM T06046 CB81CA 10489359 IC50 = 215000 nM T06046 C15IWF 10496245 Ki = 6200 nM T06046 CTN4R7 10514976 Ki = 12000 nM T06046 C56DVA 10524594 Ki = 400 nM T06046 C8MIC9 10537022 Ki = 6500 nM T06046 CDY6I3 10538489 Ki = 18000 nM T06046 C8QN6S 10540046 IC50 = 26302.68 nM T06046 C0JF6I 10575453 IC50 = 160000 nM T06046 C2X0EI 10584290 IC50 = 2000 nM T06046 CCQ8P1 10585015 IC50 = 752000 nM T06046 CJG9L3 10607934 Ki = 2700 nM T06046 C2BZ7Q 10608524 Ki = 3100 nM T06046 C1D6GY 10630840 IC50 = 39000 nM T06046 CJD2U9 10630842 IC50 = 5300 nM T06046 CZR04I 10631254 Ki = 7000 nM T06046 C9IVH2 10631255 Ki = 16000 nM T06046 C18YCZ 10632442 Ki = 1800 nM T06046 CNYF76 10634991 Ki = 2000 nM T06046 CZ7QR6 10655660 IC50 > 100000 nM T06046 C7DY3X 10656126 Ki = 17000 nM T06046 CCU7H9 10656678 Ki = 7700 nM T06046 C7R3TC 10656792 IC50 = 44000 nM T06046 C9R0NE 10680179 Ki = 1800 nM T06046 COWH50 10688427 Ki > 50000 nM T06046 C94OWI 10702801 IC50 = 21000 nM T06046 CF84US 10704325 Ki = 9000 nM T06046 C5CSV1 10727897 Ki = 9100 nM T06046 C3ON1R 10736195 Ki = 3800 nM T06046 C2KEY4 10753994 Ki = 14000 nM T06046 CL38ZM 10755655 Ki = 2800 nM T06046 CGTX82 10761718 Ki = 320 nM T06046 CM2ZI5 10773629 IC50 = 38000 nM T06046 CU5WR9 10788294 Ki = 13000 nM T06046 CGY24Z 10797080 IC50 = 39000 nM T06046 C8YXF1 10797487 Ki = 17000 nM T06046 CHNS51 10797903 Ki = 1000 nM T06046 CDW7R0 10798324 IC50 = 3065000 nM T06046 C5CE9H 10799502 IC50 = 375000 nM T06046 CS3WY5 10799675 Ki = 31000 nM T06046 CXZ1W9 10800554 Ki = 28000 nM T06046 CV2ER7 10800919 IC50 = 2200 nM T06046 C56AMX 10810281 Ki = 13000 nM T06046 C9F4GI 10822632 IC50 = 142000 nM T06046 CHND09 10823019 Ki = 14000 nM T06046 CMOE80 10825489 Ki = 17000 nM T06046 CJO21R 10845319 IC50 = 380000 nM T06046 CQ7A0W 10882498 IC50 = 14710 nM T06046 CB3CI1 10898715 IC50 = 1000 nM T06046 C93IGZ 10948273 IC50 = 54640 nM T06046 C8LVM1 10977064 IC50 = 3600 nM T06046 CN7ZJ2 11007884 IC50 = 150 nM T06046 C1WY6T 11010340 IC50 = 180 nM T06046 CTL03M 11020380 IC50 = 4600 nM T06046 C0EK3A 11034111 IC50 = 100000 nM T06046 C2MQE0 11075828 IC50 = 5000 nM T06046 C60TVY 11098403 IC50 = 100000 nM T06046 CH6Y1F 11149707 IC50 = 50000 nM T06046 C2X1GP 11161781 IC50 = 41000 nM T06046 C2BPQ8 11175135 IC50 = 2215 nM T06046 C46FGL 11210360 IC50 = 3033 nM T06046 CAWM24 11240701 IC50 = 830 nM T06046 CQV6W7 11256080 IC50 = 2930 nM T06046 CLN3E1 11267277 IC50 = 785 nM T06046 C6BM4C 11268382 IC50 = 3767 nM T06046 C5XS3F 11348978 IC50 = 12953 nM T06046 C6F7WD 11357119 IC50 > 100000 nM T06046 C8WF4O 11369870 IC50 > 100000 nM T06046 CTW93U 11390106 IC50 = 374000 nM T06046 CC98HE 11417668 IC50 = 815 nM T06046 CV97DZ 11426929 IC50 = 100000 nM T06046 C9SOQ7 11428573 IC50 = 10550 nM T06046 CIK5B2 11438569 IC50 = 13000 nM T06046 C3U6GD 11447061 IC50 = 28200 nM T06046 C0YOI9 11473924 IC50 = 12000 nM T06046 CHUP59 11481471 IC50 = 139000 nM T06046 CSBK19 11486109 IC50 = 7025 nM T06046 CP84JR 11495366 EC50 > 100000 nM T06046 C1RU2I 11496223 EC50 > 100000 nM T06046 CB43EZ 11502103 EC50 > 100000 nM T06046 CP7RX2 11523510 EC50 > 100000 nM T06046 C4JDI3 11524048 EC50 > 100000 nM T06046 CI8B3S 11531856 EC50 > 100000 nM T06046 C74RYA 11532340 EC50 > 100000 nM T06046 CO8SQ4 11532357 EC50 > 100000 nM T06046 C9F6KY 11538267 EC50 > 100000 nM T06046 CE1G4D 11539024 EC50 > 100000 nM T06046 C2KWX7 11546144 EC50 > 100000 nM T06046 CIEU85 11561546 EC50 > 100000 nM T06046 CT1Z7W 11575808 EC50 > 100000 nM T06046 CWB4J7 11582528 EC50 > 100000 nM T06046 C09EFX 11589024 EC50 > 100000 nM T06046 CBR5I2 11590027 EC50 > 100000 nM T06046 C46KUP 11596038 EC50 > 100000 nM T06046 C2KVY7 11596934 EC50 > 100000 nM T06046 C0RTF7 11609610 EC50 > 100000 nM T06046 CDC1M2 11610728 EC50 > 100000 nM T06046 CK04AC 11624646 EC50 > 100000 nM T06046 CSI50Y 11625423 EC50 > 100000 nM T06046 C9E6TG 11631971 EC50 > 100000 nM T06046 C0MHE1 11633531 EC50 > 100000 nM T06046 CWG4J9 11639946 EC50 > 100000 nM T06046 CL7Q3I 11646432 EC50 > 100000 nM T06046 C4F0CK 11646596 EC50 > 100000 nM T06046 CA6D9Z 11654166 EC50 > 100000 nM T06046 C8UJ1K 11695590 EC50 > 100000 nM T06046 CM7YA3 11703771 EC50 > 100000 nM T06046 C5I6PB 11744927 IC50 = 4000 nM T06046 CQ5RJ9 11957582 IC50 = 78000 nM T06046 CG63IC 12109769 IC50 > 100000 nM T06046 CS5D0P 12404013 IC50 = 600 nM T06046 CLVQ03 12449028 IC50 > 100000 nM T06046 C2NX4W 12709336 IC50 > 50000 nM T06046 CNJ76X 12778905 IC50 = 93000 nM T06046 C4XK7S 12778908 IC50 = 600 nM T06046 CEJ53H 12778910 IC50 = 15000 nM T06046 CO7T1N 12969094 IC50 = 50000 nM T06046 CXA84F 13196077 IC50 > 50000 nM T06046 CZ2D9G 13268358 Ki = 26000 nM T06046 C9D4CW 13302397 IC50 = 16600 nM T06046 C9MC3D 13768254 IC50 = 53703.18 nM T06046 CI07KP 13768262 IC50 > 100000 nM T06046 CZK9A7 15287360 IC50 = 3400 nM T06046 C96DOX 15381020 IC50 = 40000 nM T06046 CSJ32F 15453846 IC50 = 58000 nM T06046 C0O5LD 15453847 IC50 = 3000 nM T06046 CAJF09 15512769 IC50 = 448 nM T06046 CHR3S4 15512781 IC50 = 685 nM T06046 CPF1W0 15871186 IC50 = 24000 nM T06046 COV8E5 15887952 IC50 = 660000 nM T06046 C2ZYA6 15951338 IC50 = 6240 nM T06046 CL0SF3 15951408 IC50 = 17500 nM T06046 C1Q8IV 15951410 IC50 = 19000 nM T06046 C6Z1DA 16739325 IC50 = 1600 nM T06046 CD3CT0 17793169 IC50 = 458000 nM T06046 C9V0XQ 17897120 IC50 = 578000 nM T06046 C3X9JP 17958630 IC50 = 48140 nM T06046 CP2D3I 18356525 Ki > 50000 nM T06046 C6RA2L 18414528 IC50 = 372 nM T06046 CKMV50 18428554 IC50 = 13000 nM T06046 CMSA79 18687946 Ki = 33000 nM T06046 C05KOC 18721714 IC50 > 50000 nM T06046 CY28GR 18721729 IC50 > 50000 nM T06046 CS76LE 18785786 IC50 = 8000 nM T06046 C4EOC0 18785787 IC50 = 280 nM T06046 CYX62M 18785788 IC50 = 100000 nM T06046 CV37DL 18785796 IC50 = 55000 nM T06046 CH4QG0 18785802 IC50 = 10000 nM T06046 CG8ZV1 18785805 IC50 = 750 nM T06046 CHBN50 18785824 IC50 = 1900 nM T06046 CCM32F 18785825 IC50 = 900 nM T06046 C80CGE 18785840 IC50 = 4000 nM T06046 C1JMD3 18785851 IC50 = 40000 nM T06046 CRZ4G5 18785857 IC50 = 19000 nM T06046 CH26IT 18785878 IC50 = 80 nM T06046 C3W6ZT 18785879 IC50 = 6000 nM T06046 CZ0F5Y 18785885 IC50 = 5000 nM T06046 CFLJ71 18785905 IC50 = 44000 nM T06046 C1U9RA 18785910 IC50 = 5000 nM T06046 CH3T2Z 18785914 IC50 = 86000 nM T06046 CI8Z7F 18785933 IC50 = 120 nM T06046 C10PZK 18785936 IC50 = 9000 nM T06046 CTEZ46 18785938 IC50 = 9500 nM T06046 CY7EO4 18800758 IC50 = 2920000 nM T06046 CW0IX3 18983434 IC50 = 53000 nM T06046 CFB10N 20102781 IC50 = 13600 nM T06046 CQZ84B 21192814 IC50 = 2500 nM T06046 CN5A8J 21834414 IC50 = 19800 nM T06046 CW2VK6 21878467 IC50 = 2900 nM T06046 CH70CD 22133392 IC50 > 100000 nM T06046 CZ3X6F 24745386 Ki > 50000 nM T06046 CBNT78 24745536 Ki = 43000 nM T06046 CN1D9J 24758920 IC50 = 6330 nM T06046 CPH67W 24764596 Ki = 20000 nM T06046 C02RPF 24782142 EC50 > 100000 nM T06046 C2UR8E 24782146 EC50 > 100000 nM T06046 C74IOP 24782646 EC50 = 5800 nM T06046 C40NIF 24782649 EC50 > 100000 nM T06046 CD2T4M 24782902 EC50 > 100000 nM T06046 CFG23E 24782903 EC50 = 6800 nM T06046 CM50WK 24785172 EC50 = 1600 nM T06046 C6U0PV 24785174 EC50 = 1300 nM T06046 CD7K3S 24785426 EC50 > 100000 nM T06046 CT2UV6 24785697 EC50 > 100000 nM T06046 C3MWU8 24785698 EC50 > 100000 nM T06046 CWK68M 24785700 EC50 = 5900 nM T06046 C4TC8F 24785702 EC50 > 100000 nM T06046 CO65CH 24785966 EC50 > 100000 nM T06046 CTLA48 24785968 EC50 = 1300 nM T06046 C5VBE0 24787679 IC50 = 4000000 nM T06046 CPN5Z3 24798097 Ki = 85.2 nM T06046 C86KAI 24798098 Ki = 26000 nM T06046 C7IXF0 24850786 Ki = 416.7 nM T06046 CFJX70 24850913 Ki = 366.6 nM T06046 CPQ15V 24894148 IC50 = 4900 nM T06046 CYU1V8 24894149 IC50 > 100000 nM T06046 CNX5Q3 24894150 IC50 > 100000 nM T06046 C3QK6V 24894151 IC50 > 100000 nM T06046 C6J0NK 24894153 IC50 = 80 nM T06046 C7Q3YX 24894154 IC50 = 200 nM T06046 C4Z3KW 24941263 IC50 = 200 nM T06046 C7DM6Y 25021186 Ki = 95.2 nM T06046 CR3I9Y 25050394 EC50 = 34000 nM T06046 C39DOQ 25050395 EC50 = 37000 nM T06046 CW0Q3F 25210996 EC50 = 8800 nM T06046 C9T1XJ 25211376 EC50 > 100000 nM T06046 CD09PR 25211378 EC50 > 100000 nM T06046 CD0F1I 25211400 IC50 = 8300 nM T06046 C5K3ZC 25211401 IC50 = 7100 nM T06046 C9O3QC 25211403 IC50 = 12000 nM T06046 CSG69X 25211404 IC50 = 11000 nM T06046 CF79GW 25211493 EC50 > 100000 nM T06046 CE9DK7 25211494 EC50 > 100000 nM T06046 C0DOS1 25211596 EC50 > 100000 nM T06046 CT3ID6 25211597 EC50 > 100000 nM T06046 C2UQJ6 25211598 EC50 = 39000 nM T06046 C43HVC 25211599 EC50 > 100000 nM T06046 CDV7E8 25211804 EC50 > 100000 nM T06046 CKI86X 25211805 EC50 = 26000 nM T06046 CHW2X0 25211910 EC50 = 16500 nM T06046 CW0Q7Y 25212125 IC50 = 6400 nM T06046 C4EF2A 25212418 IC50 = 13000 nM T06046 C7ESB2 25231661 IC50 = 80000 nM T06046 CJ92GL 25231666 IC50 = 90000 nM T06046 CCO21E 25231830 IC50 = 300000 nM T06046 CNV40T 42618036 EC50 > 100000 nM T06046 CH7AS5 42618037 EC50 > 100000 nM T06046 C97FDE 42618038 EC50 > 100000 nM T06046 C3MJQ4 42618039 EC50 > 100000 nM T06046 C1YO7H 42618040 EC50 = 26000 nM T06046 C0B6JO 42618041 EC50 > 100000 nM T06046 C20NYG 42618042 EC50 = 15000 nM T06046 C3G6HZ 42618043 EC50 > 100000 nM T06046 C3C4FA 42618044 EC50 > 100000 nM T06046 C2SK5R 42618045 EC50 > 100000 nM T06046 CI9PO8 42618046 EC50 > 100000 nM T06046 C1V0KI 42618047 EC50 > 100000 nM T06046 CXE5C2 42618048 EC50 = 13000 nM T06046 C3S4NL 42618049 EC50 = 41000 nM T06046 CN6WQ5 42618050 EC50 > 100000 nM T06046 C5F6PW 42618052 EC50 = 6800 nM T06046 CMQI75 42618053 EC50 > 100000 nM T06046 CN34WV 42618054 EC50 > 100000 nM T06046 CH81PY 42618060 EC50 > 100000 nM T06046 C4QS7B 42618062 EC50 > 100000 nM T06046 CAZ25X 42618063 EC50 = 33000 nM T06046 CX5NI3 42618064 EC50 > 100000 nM T06046 C54TBN 42618065 EC50 > 100000 nM T06046 C0I4MK 42618066 EC50 = 3000 nM T06046 CGU3N8 42618068 EC50 = 420 nM T06046 C5UN1C 42618069 EC50 = 1200 nM T06046 C8JFX2 42618070 EC50 = 35000 nM T06046 CRQ96D 42634153 IC50 = 40300 nM T06046 CS0DX1 44264963 IC50 = 12000 nM T06046 C9C5TH 44294245 Ki = 8800 nM T06046 CKT5C3 44294421 Ki = 39000 nM T06046 CYI6D2 44302109 IC50 = 3300 nM T06046 CE9LX0 44302114 IC50 = 9600 nM T06046 CR5C8Z 44302148 IC50 = 52000 nM T06046 C1T7UQ 44302150 IC50 = 8700 nM T06046 C3R1FC 44313302 IC50 = 31000 nM T06046 CHD4J9 44313313 IC50 = 580 nM T06046 CWN2P5 44313352 IC50 = 7400 nM T06046 C2OAM9 44313353 IC50 = 360 nM T06046 C27LBK 44313364 IC50 = 510 nM T06046 CRL32W 44313509 IC50 = 520 nM T06046 C0NUT2 44313550 IC50 = 240 nM T06046 CWR7G1 44313551 IC50 = 320 nM T06046 C2YDZ6 44319656 IC50 = 2300 nM T06046 CQYW59 44319709 IC50 = 14000 nM T06046 CO1Z2F 44319710 IC50 = 20000 nM T06046 C54VXO 44319711 IC50 = 4100 nM T06046 CA81IQ 44319778 IC50 = 12000 nM T06046 CD1QB5 44319779 IC50 = 960 nM T06046 CR3HT4 44319780 IC50 = 21000 nM T06046 C59RGW 44319825 IC50 = 2300 nM T06046 C76IJF 44319826 IC50 = 6200 nM T06046 CY8K0G 44319828 IC50 = 24000 nM T06046 CQ5A4R 44320031 IC50 = 54000 nM T06046 C0PQ4L 44320069 IC50 > 200000 nM T06046 CL42AK 44320084 IC50 = 57000 nM T06046 CV4XW8 44320115 IC50 > 200000 nM T06046 CHT83A 44320347 IC50 = 825 nM T06046 C80ORG 44322605 IC50 = 709000 nM T06046 CCM47P 44328869 Ki = 1900 nM T06046 CZ2BS4 44328871 Ki = 9100 nM T06046 C7FG5O 44328879 Ki = 46000 nM T06046 C4N5IJ 44328899 Ki = 8000 nM T06046 C34CQV 44328929 Ki = 17000 nM T06046 C0BDZ8 44328932 Ki = 44000 nM T06046 CSG52F 44328934 Ki = 14000 nM T06046 CDF12B 44328946 Ki > 50000 nM T06046 CVO68P 44328955 Ki = 39000 nM T06046 CTAF63 44328957 Ki > 50000 nM T06046 C0W1JK 44328968 Ki = 15000 nM T06046 C7GS5O 44328973 Ki > 50000 nM T06046 C14UCS 44328998 Ki > 50000 nM T06046 CEP9D7 44329003 Ki = 38000 nM T06046 CZQ78B 44329038 Ki = 17000 nM T06046 CG6F2P 44329061 Ki = 27000 nM T06046 C8UEJ6 44329070 Ki = 7900 nM T06046 C39GJB 44329072 Ki > 50000 nM T06046 CPOB75 44329074 Ki > 50000 nM T06046 C3OUZ7 44329119 Ki = 36000 nM T06046 CMW2I5 44329128 Ki = 27000 nM T06046 CNZ5T9 44329167 Ki = 46000 nM T06046 CP4ZU0 44329169 Ki > 50000 nM T06046 CW1VT4 44329187 Ki > 50000 nM T06046 C7PG5J 44329191 Ki > 50000 nM T06046 C1TKS5 44329193 Ki > 50000 nM T06046 C86AGM 44329195 Ki = 13000 nM T06046 C25XJI 44329227 Ki = 9500 nM T06046 CV67AL 44329240 Ki > 50000 nM T06046 CEBZ52 44329255 Ki = 3000 nM T06046 CYX4T3 44329820 IC50 > 50000 nM T06046 C1FHY4 44329948 IC50 = 20300 nM T06046 C81QDL 44329949 IC50 = 8400 nM T06046 C5W4FL 44329963 IC50 = 15500 nM T06046 CBQ1O0 44329995 IC50 = 15900 nM T06046 C8F5EQ 44341087 IC50 = 2930000 nM T06046 CQ0CU9 44341212 IC50 = 4800 nM T06046 CU62NQ 44341315 IC50 = 930000 nM T06046 CWQ18O 44341316 IC50 = 695000 nM T06046 C2YC1E 44347417 IC50 = 212000 nM T06046 C86PTS 44347432 IC50 = 23600 nM T06046 CQ6DG0 44370661 IC50 > 100000 nM T06046 C0FRX8 44370662 IC50 > 100000 nM T06046 C46TVU 44370689 IC50 > 100000 nM T06046 CYI91R 44370690 IC50 > 100000 nM T06046 C9GZB5 44370704 IC50 > 100000 nM T06046 CKQ20Y 44370705 IC50 = 72000 nM T06046 CS4M3D 44370729 IC50 > 1000000 nM T06046 CI7K3E 44370730 IC50 > 100000 nM T06046 C6VS9A 44370736 IC50 = 155000 nM T06046 C12SON 44370747 IC50 = 13000 nM T06046 CF5W2Z 44377082 IC50 = 22000 nM T06046 CW0F6J 44377099 IC50 = 38000 nM T06046 C7K8XO 44377152 IC50 = 66000 nM T06046 C6C2YV 44377153 IC50 = 14000 nM T06046 C2NZ1X 44393481 IC50 > 50000 nM T06046 CDSJ39 44393485 IC50 > 50000 nM T06046 C10WEK 44393495 IC50 > 50000 nM T06046 C3GDF7 44393630 IC50 = 16500 nM T06046 C9M5SP 44393639 IC50 > 32000 nM T06046 C6CDT1 44393666 IC50 > 32000 nM T06046 CTD27K 44393700 IC50 > 7700 nM T06046 CJ02FD 44393705 IC50 = 21943 nM T06046 C93KUZ 44393711 IC50 > 32000 nM T06046 C85GFC 44396192 IC50 > 50000 nM T06046 C4XL3B 44399796 IC50 = 4500 nM T06046 C53KME 44399834 IC50 > 5000 nM T06046 CU98HN 44399945 IC50 = 2000 nM T06046 CYW0O2 44400067 IC50 = 15300 nM T06046 CU6M4D 44402389 IC50 > 1000000 nM T06046 C94GAW 44402453 IC50 > 1000000 nM T06046 CDIR71 44402600 IC50 = 11000 nM T06046 CQTC93 44402628 IC50 > 1000000 nM T06046 CL5I8G 44430315 IC50 = 9400 nM T06046 CEH14S 44430628 IC50 = 6000 nM T06046 C0WX4U 44430629 IC50 = 12000 nM T06046 CUO30Z 44430631 IC50 = 16000 nM T06046 C90QJT 44430632 IC50 = 13000 nM T06046 CLZ51V 44430633 IC50 = 8000 nM T06046 CWT98D 44430634 IC50 = 700 nM T06046 C62UWN 44430635 IC50 = 2100 nM T06046 CI8WV0 44430636 IC50 = 16000 nM T06046 CG13ZP 44430637 IC50 = 3800 nM T06046 C43QST 44430638 IC50 = 5700 nM T06046 C8PTS2 44430640 IC50 = 5200 nM T06046 C58QXR 44430641 IC50 = 59000 nM T06046 C4PE7R 44455626 IC50 = 4000 nM T06046 C1E3AV 44455627 IC50 = 4400 nM T06046 C4UZH5 44455631 IC50 = 983 nM T06046 C34XKU 44455663 IC50 = 2100 nM T06046 C50IWU 44455685 IC50 = 570 nM T06046 C9E7NX 44455718 IC50 = 220 nM T06046 CH9W2F 44455719 IC50 = 1000 nM T06046 CG6I8D 44455720 IC50 = 1700 nM T06046 CV8JE9 44455746 IC50 = 540 nM T06046 CEGL71 44455747 IC50 = 860 nM T06046 C8DQV4 44455748 IC50 = 4300 nM T06046 CHAZ31 44455749 IC50 = 680 nM T06046 CPDZ45 44455769 IC50 = 450 nM T06046 C02SZW 44455770 IC50 = 1100 nM T06046 CQ2VA3 44455771 IC50 = 1100 nM T06046 C6CYN7 44455794 IC50 = 820 nM T06046 CVMY02 44455795 IC50 = 810 nM T06046 CN3D9Q 44455797 IC50 = 1400 nM T06046 CSIX74 44455821 IC50 = 770 nM T06046 C03BYA 44565909 EC50 = 6100 nM T06046 C8DUG3 44566070 EC50 = 2500 nM T06046 CB1Y8N 49796134 IC50 = 2420000 nM T06046 CN8T5X 49796514 IC50 = 1980000 nM T06046 CB29CM 49797485 IC50 = 20000 nM T06046 CM2D5Z 49836940 EC50 = 15000 nM T06046 CZ51GS 49836941 EC50 > 100000 nM T06046 CM2JB5 49836942 EC50 = 4200 nM T06046 C6ZA7M 49836943 EC50 = 11300 nM T06046 C1IHW8 49836944 EC50 = 6800 nM T06046 CM10KE 49837060 EC50 = 3900 nM T06046 C3J2SH 49837061 EC50 = 2900 nM T06046 CP92KI 49837062 EC50 = 21000 nM T06046 C2ZD0V 49837063 EC50 > 100000 nM T06046 C1SB6T 49837065 EC50 = 13000 nM T06046 CK38CR 49837066 EC50 = 9200 nM T06046 CD8GN9 49837170 EC50 > 100000 nM T06046 CZJ85F 49864405 IC50 = 50000 nM T06046 C1MYW7 53233132 IC50 = 15000 nM T06046 CZWO31 53387025 IC50 = 45600 nM T06046 C6AYE3 53392451 IC50 = 14300 nM T06046 CQ8W0K 54580275 IC50 = 2400 nM T06046 C6TN1Y 54583301 IC50 > 100000 nM T06046 C6QK1A 56593711 IC50 = 7100 nM T06046 CXSQ19 56593712 IC50 = 26500 nM T06046 CY70WM 56593713 IC50 = 10700 nM T06046 C48VIC 56593714 IC50 = 46200 nM T06046 C4U6BD 56593857 IC50 = 23300 nM T06046 CC86JF 56659406 IC50 = 1071.52 nM T06046 CSBN93 56659435 IC50 > 100000 nM T06046 C6P5YB 56666339 IC50 > 100000 nM T06046 CDF86T 56669739 IC50 = 87096.36 nM T06046 CRZ08C 56673237 IC50 = 204173.79 nM T06046 C8TA3D 56679900 IC50 > 100000 nM T06046 C73MZW 56924689 IC50 = 195000 nM T06046 C83REA 56949933 IC50 = 109000 nM T06046 C2DJ7A 56949934 IC50 = 84800 nM T06046 C3B4DI 56949935 IC50 = 21500 nM T06046 C5DK8C 56950062 IC50 = 7120 nM T06046 C13TGD 56950064 IC50 = 3360 nM T06046 CF2VW1 56950067 IC50 = 7170 nM T06046 CHO6F5 56950186 IC50 = 99000 nM T06046 CHQ5S6 56950187 IC50 = 243000 nM T06046 CRG42P 56950331 IC50 = 220000 nM T06046 C6BZ7V 56951568 IC50 = 1500 nM T06046 C0UW5Z 57341142 IC50 = 33300 nM T06046 CS2FH5 57341143 IC50 = 63900 nM T06046 C2AUM9 57341144 IC50 = 40700 nM T06046 CX1FQ0 57341332 IC50 = 22500 nM T06046 CN3Y9D 57341333 IC50 = 46500 nM T06046 C3H1GV 57341334 IC50 = 30200 nM T06046 C0Z3JI 57341335 IC50 = 32900 nM T06046 C83DHY 57341336 IC50 = 23500 nM T06046 CDU9W0 57341337 IC50 = 39200 nM T06046 CBO89M 57384807 IC50 = 47100 nM T06046 C2BAZ9 57385041 IC50 = 32000 nM T06046 C2TAS4 57385549 IC50 = 7760 nM T06046 CX2TG9 57385550 IC50 = 77600 nM T06046 CVM67R 57385790 IC50 = 11000 nM T06046 COQ83X 57391112 EC50 > 100000 nM T06046 C19RIY 57391700 IC50 = 14000 nM T06046 CB1NH9 57392807 EC50 > 100000 nM T06046 C6FD9C 57393301 IC50 = 7500 nM T06046 C6HO3K 57393302 IC50 > 30000 nM T06046 C01NAX 57393303 IC50 > 30000 nM T06046 C7TM3R 57393317 IC50 > 30000 nM T06046 C6RKY7 57393439 IC50 = 79000 nM T06046 C5QMZ6 57393919 IC50 = 650 nM T06046 C21UDR 57394528 EC50 > 100000 nM T06046 CVC7Z2 57394614 EC50 > 100000 nM T06046 CPQ0S7 57394615 EC50 > 100000 nM T06046 C9J6IM 57395031 IC50 > 30000 nM T06046 CP4TV8 57395168 IC50 > 30000 nM T06046 COKU75 57396367 EC50 > 100000 nM T06046 CV7HI9 57396371 EC50 > 100000 nM T06046 CL0P6T 57396785 IC50 = 11000 nM T06046 C2QS6D 57396941 IC50 = 5500 nM T06046 C4BO9G 57398563 IC50 = 8300 nM T06046 CAY3X7 57398682 IC50 > 30000 nM T06046 C1DCN7 57401588 EC50 > 100000 nM T06046 CQ5HU7 57401590 EC50 > 100000 nM T06046 CI2DY9 57403339 EC50 > 100000 nM T06046 CD9P4Z 57403764 IC50 > 30000 nM T06046 C2ONF1 57403909 IC50 = 23000 nM T06046 CYQ70T 57403910 IC50 = 21000 nM T06046 CM6C1O 57403911 IC50 = 13000 nM T06046 CSWV56 57474449 IC50 = 64700 nM T06046 C0L5HT 62706594 IC50 = 4740 nM T06046 CJHB32 62706595 IC50 = 17000 nM T06046 C9EIX4 62706596 IC50 = 4040 nM T06046 C04WBM 62706597 IC50 = 8000 nM T06046 CS9KV1 62706598 IC50 = 28700 nM T06046 CX72ZW 62706764 IC50 = 29500 nM T06046 C24YCI 62706765 IC50 = 117000 nM T06046 CEL48Q 62706766 IC50 > 100000 nM T06046 C7XEA4 62706767 IC50 = 37100 nM T06046 CC5B6H 62706768 IC50 = 47100 nM T06046 CO7AH9 66912415 IC50 = 11200 nM T06046 CA7DI2 66912425 IC50 = 10200 nM T06046 C2PK8Q 66912454 IC50 = 17100 nM T06046 C37DOA 66912484 IC50 = 19100 nM T06046 C78AWC 66912498 IC50 = 23300 nM T06046 C8Y7AV 66912516 IC50 = 11800 nM T06046 CPB9C5 66912809 IC50 = 34000 nM T06046 CF0J3M 67340183 IC50 = 6000 nM T06046 C5HSI6 67492912 IC50 = 415000 nM T06046 C9FMX2 67493358 IC50 = 99100 nM T06046 C3UO2F 70686000 IC50 = 49300 nM T06046 CWO02R 70688127 IC50 = 32000 nM T06046 C0M6DH 71484435 IC50 = 4080 nM T06046 CIE6A1 71486265 IC50 = 4070 nM T06046 C2Y1CX 71486266 IC50 = 410 nM T06046 CO8D6C 71486267 IC50 = 770 nM T06046 CS0X2Q 71486405 IC50 = 1580 nM T06046 C7DH8X 71486406 IC50 = 4670 nM T06046 C9VIN3 71486407 IC50 = 1090 nM T06046 CRZ73J 71486408 IC50 = 52200 nM T06046 CW9V2Q 71718237 IC50 = 3500 nM T06046 CC6Q5R 72771081 Ki = 11800 nM T06046 C0TSY5 72771082 Ki = 9490 nM T06046 CXZ71D 76033629 IC50 = 68900 nM T06046 C26ADC 90662876 IC50 = 24500 nM T06046 C3QU2O 90662877 IC50 = 16000 nM T06046 CYUW16 90664333 IC50 = 18900 nM T06046 CRK93Y 90664334 IC50 = 3150 nM T06046 CAUK54 90664335 IC50 = 9200 nM T06046 CR35FV 90664340 IC50 = 29800 nM T06046 CZ8H2M 90664341 IC50 = 24500 nM T06046 C5UNM2 90664342 IC50 = 22400 nM T06046 CE5H8T 90664346 IC50 = 66200 nM T06046 CVY3L6 90664347 IC50 = 75000 nM T06046 CPNS27 90664349 IC50 = 317000 nM T06046 C5RHW1 90664461 IC50 = 12100 nM T06046 CRX47I 90664467 IC50 = 249000 nM T06046 CNLO43 90664468 IC50 = 43000 nM T06046 C2G0XJ 90664469 IC50 = 36100 nM T06046 CU7Q9V 90664588 IC50 = 23000 nM T06046 C9TLX0 90664602 IC50 = 4490 nM T06046 C7JIW4 90664606 IC50 = 27500 nM T06046 CP1JM7 90664607 IC50 = 65300 nM T06046 CN7P3V 90664608 IC50 = 82200 nM T06046 C8LFX7 90664695 IC50 = 24000 nM T06046 CU29TX 90664696 IC50 = 30600 nM T06046 C7FQ5W 90664698 IC50 = 28300 nM T06046 C8X1LA 90664704 IC50 = 13900 nM T06046 C1PHN4 90664711 IC50 = 15000 nM T06046 C6EGO9 90664714 IC50 = 8720 nM T06046 CS65XI 90664715 IC50 = 3700 nM T06046 CJ61NW 90664716 IC50 = 1920 nM T06046 CQT69X 90664721 IC50 = 58700 nM T06046 CVXO58 90664722 IC50 = 64400 nM T06046 CUNK69 90664723 IC50 = 9500 nM T06046 CE7H6D 90664727 IC50 = 97400 nM T06046 C9Y2FD 90664833 IC50 = 19000 nM T06046 CE3RV1 90664839 IC50 = 73600 nM T06046 CGK56Q 90664840 IC50 = 25200 nM T06046 C0JM7D 90664841 IC50 = 154000 nM T06046 CL0TG4 90664842 IC50 = 24300 nM T06046 CN3A1P 90664848 IC50 = 36100 nM T06046 C7H8FN 90664849 IC50 = 56300 nM T06046 CA81EW 90664850 IC50 = 20000 nM T06046 C7HGP1 90664855 IC50 = 60500 nM T06046 C8F7HI 90664950 IC50 = 2530 nM T06046 CHA2T6 90664963 IC50 = 6400 nM T06046 CJ01LW 90664969 IC50 = 41100 nM T06046 C8PCH5 90664970 IC50 = 194000 nM T06046 CYT2F5 90664975 IC50 = 105200 nM T06046 CG78YO 90665018 IC50 = 3500 nM T06046 C5FZK7 90665071 IC50 = 37700 nM T06046 CF14BZ 90665089 IC50 = 15800 nM T06046 CI4H7Y 90665090 IC50 = 3800 nM T06046 C7PHT4 90665099 IC50 = 24200 nM T06046 C0LM7T 90665100 IC50 = 30800 nM T06046 CY4F6W 90665101 IC50 = 47100 nM T06046 C57NEK 90665196 IC50 = 11500 nM T06046 C3E6MO 90665203 IC50 = 12400 nM T06046 C79CZW 90665204 IC50 = 3370 nM T06046 C2WUY8 90665205 IC50 = 650 nM T06046 CK62BX 90665207 IC50 = 42700 nM T06046 C02PLA 90665208 IC50 = 119000 nM T06046 CB63ER 90665216 IC50 = 22400 nM T06046 CQ35RI 91971384 Ki = 17300 nM T06046 CB0A4F 91971388 Ki = 7410 nM T06046 C6JP8E 119057273 Ki = 73006 nM T06046 C1MFO5 119057274 Ki = 22536 nM T06046 COLQ09 119081686 Ki = 42563 nM T06046 CL3DK1 119081688 Ki = 22895 nM T06046 CUD7Q0 119081689 Ki = 39533 nM T06046 CL98KI 121250394 Ki = 1030 nM T06046 CZM87C 121250396 Ki = 2080 nM T06046 CEA5V4 121250401 Ki = 5790 nM T06046 C6EH9G 121250403 Ki = 2700 nM T06046 CTQ9U6 121250406 Ki = 5760 nM T06046 CH7Q5A 124136836 Ki = 6660 nM T06046 CG0EN1 124136841 Ki = 15000 nM T06046 CF70JE 124136845 Ki = 18900 nM T06046 CRPM16 124136846 Ki = 6090 nM T06046 C7JLU1 124136856 Ki = 21000 nM T06046 CD24UM 124136858 Ki = 4800 nM T06046 CLZ38Y 124136872 Ki = 16100 nM T06046 CG0HT3 124136874 Ki = 4190 nM T06046 CP95UD 124136876 Ki = 12300 nM T06046 CHOG43 124136880 Ki = 6080 nM T06046 C8E1MD 124136896 Ki = 43000 nM T06046 C7ONE0 124136898 Ki = 5040 nM T06046 CT2PQ8 124136901 Ki = 22100 nM T06046 CH5GX6 124145845 Ki = 1580 nM T06046 CS9E0R 127050046 Ki = 18271 nM T06046 CL2YX7 130449136 Ki = 39505 nM T06046 C1UTC8 130449148 Ki = 20117 nM T06046 CTL8B5 130449158 Ki = 83976 nM T06046 CV41FA 130449315 Ki = 20816 nM T06046 C7J9BX 134686794 Ki = 42086 nM T06046 C6OGU3 134686796 Ki = 8668 nM T06046 C0A9BD 134686797 Ki = 68539 nM T06046 CGX96C 134686798 Ki = 19415 nM T06046 C76NBO 135409922 IC50 = 4120 nM T06046 C83ZLX 135449023 IC50 = 10050 nM T06046 C7O9XT 135458572 IC50 > 100000 nM T06046 C5H2QR 135674618 IC50 > 500000 nM T06046 C8MN2E 135973134 IC50 = 253000 nM T06046 CMCS36 136035301 IC50 = 253200 nM T06046 CPC52T 136035302 IC50 > 500000 nM T06046 COA8D6 136109078 IC50 > 500000 nM T06046 CHC62Q 136109080 IC50 = 350700 nM T06046 CB4UO8 136109082 IC50 = 208600 nM T06046 CL41DA 137530114 Ki = 35028 nM T06046 C9USH3 137530118 Ki = 50280 nM T06046 CDKB20 137530119 Ki = 16960 nM T06046 CSR3F0 137530120 Ki = 35758 nM T06046 CA39SN 137530121 Ki = 25548 nM T06046 CH1S5L 137530126 Ki = 21980 nM T06046 CDOS52 137633546 Ki = 51542 nM T06046 C95OYQ 137637529 Ki = 69888 nM T06046 CAN9G4 146025971 Ki = 18200 nM T06046 CMTI65 146025972 Ki = 12900 nM T06046 CN6H0M 146025973 Ki = 20200 nM T06046 CQ9P2B 146025974 Ki = 22800 nM T06046 CN8JM9 146025975 Ki = 21000 nM T06046 CYOA91 146025976 Ki = 23700 nM T06046 CS0BW8 146025977 Ki = 7730 nM T06046 CY37WD 146025978 Ki = 6200 nM T06046 C4S1ZP 146025979 Ki = 27300 nM T06046 C8RWQ4 146025980 Ki = 20000 nM T06046 C9R5SN 146025981 Ki = 8310 nM T06046 CCP8X4 155513324 Ki = 41900 nM T06046 CG35TK 155527043 Ki = 23300 nM T06046 CF85SO 155534420 Ki = 5650 nM T06046 C7ZTA4 155540835 Ki = 52600 nM T06046 COAM39 155543079 Ki = 18700 nM T06046 D00EVC 10197851 IC50 = 150 nM T06046 D00KOE 18983431 IC50 = 87800 nM T06046 D00TDJ 44430622 IC50 = 12000 nM T06046 D01EHS 15552206 IC50 = 5000 nM T06046 D01ILO 15689 IC50 = 1100 nM T06046 D01MEA 22617750 IC50 = 77000 nM T06046 D01RGM 3311 Ki = 9400 nM T06046 D01TDG 347590 Ki = 400 nM T06046 D01XOR 44396191 IC50 = 6000 nM T06046 D01YNT 10012278 IC50 = 205900 nM T06046 D02ELA 107984 Ki = 810 nM T06046 D02EOF 10725313 IC50 = 14500 nM T06046 D02MFQ 10606829 IC50 = 90000 nM T06046 D02TMX 9855524 IC50 = 50 nM T06046 D02TYS 44396204 IC50 = 10500 nM T06046 D03CAJ 10375155 IC50 = 2770 nM T06046 D03FJM 10198326 IC50 = 500 nM T06046 D03JXX 10261068 IC50 = 600 nM T06046 D03ODQ 15463448 IC50 = 25000 nM T06046 D03QMU 10104379 IC50 = 102500 nM T06046 D03QSQ 19049087 IC50 = 227000 nM T06046 D03WOZ 1893 IC50 = 36000 nM T06046 D04QFO 44393534 IC50 > 50000 nM T06046 D05APC 19049123 IC50 = 3500 nM T06046 D05PZA 25231659 IC50 = 350000 nM T06046 D05VAB 9886249 IC50 > 100000 nM T06046 D06VYU 10198539 IC50 = 1000 nM T06046 D07BLJ 44322961 IC50 = 186300 nM T06046 D07INO 18428457 IC50 = 24000 nM T06046 D07MFH 44323014 IC50 = 247800 nM T06046 D07OQX 9812839 IC50 > 50000 nM T06046 D07PYV 10439 IC50 = 2800 nM T06046 D07VFC 42625451 IC50 = 1500 nM T06046 D08ALG 9793728 IC50 = 15250 nM T06046 D08CMQ 18721725 IC50 = 60000 nM T06046 D08FXW 42625617 IC50 = 1428 nM T06046 D08ISP 19049152 IC50 = 104000 nM T06046 D08JSR 3287412 IC50 = 87000 nM T06046 D08PZX 15463450 IC50 = 50000 nM T06046 D08WEI 18721726 IC50 = 5000 nM T06046 D09BKV 15463449 IC50 = 50000 nM T06046 D09NRX 18721724 IC50 = 1100 nM T06046 D0AO5D 1433 Ki = 75000 nM T06046 D0C1OB 12778904 IC50 = 4600 nM T06046 D0D0TO 85237 IC50 = 4700 nM T06046 D0D2WC 17892465 IC50 = 5500 nM T06046 D0D3CJ 10308091 IC50 = 112201.85 nM T06046 D0D7PK 3268009 IC50 = 146 nM T06046 D0D9LT 12778906 IC50 = 1900 nM T06046 D0DI7W 9793827 IC50 = 230 nM T06046 D0G4ZL 19049163 IC50 = 8700 nM T06046 D0I3ZP 44396203 IC50 = 450 nM T06046 D0I7VD 5139 IC50 = 1300 nM T06046 D0IR4Y 9995251 IC50 = 39070 nM T06046 D0J2RI 19049061 IC50 = 60600 nM T06046 D0J7NS 15887953 IC50 = 2600 nM T06046 D0K1CM 10749191 IC50 = 58900 nM T06046 D0K4SV 4102304 IC50 = 85000 nM T06046 D0K4YY 44399940 IC50 = 5500 nM T06046 D0L9SL 44322997 IC50 = 1363000 nM T06046 D0LB9U 44322572 IC50 = 49300 nM T06046 D0LE6N 19049158 IC50 = 4700 nM T06046 D0M4BM 23042899 IC50 = 8200 nM T06046 D0N3HU 15463447 IC50 = 43600 nM T06046 D0N8EU 173566 IC50 = 5900 nM T06046 D0O3XZ 1533 IC50 = 72 nM T06046 D0O9II 189081 IC50 = 7100 nM T06046 D0OW8M 9797857 IC50 > 100000 nM T06046 D0R9KX 44399941 IC50 = 12500 nM T06046 D0S7MJ 25231669 IC50 = 300000 nM T06046 D0SB5H 18721719 IC50 = 4100 nM T06046 D0VN7G 44393480 IC50 = 33000 nM T06046 D0W9UV 21507 IC50 = 170 nM T06046 D0X2XQ 10467406 IC50 = 9200 nM T06046 D0X6MB 9942127 IC50 = 1800 nM T06046 D0X6QY 19049121 IC50 = 6300 nM T06046 D0XJ1C 10396852 IC50 = 520 nM T06046 D0Y8DZ 10130105 IC50 = 1500 nM T04820 D09EGZ 2719 IC50 = 150000 nM T04820 D0GQ7K 4046 IC50 = 12000 nM T04820 D03KKR 3547 IC50 > 500000 nM T04820 D05ADP 160355 IC50 > 1000000 nM T04820 D0E3TC 44259 IC50 = 4000 nM T04820 D0L4FS 5280961 IC50 = 93000 nM T04820 D00PWQ 3820 IC50 = 15000 nM T04820 D00BPA 4592 IC50 = 1100000 nM T04820 C32LCX 3545 IC50 > 500000 nM T04820 CA47TS 3546 IC50 > 500000 nM T04820 CWT4N9 4216 IC50 > 500000 nM T04820 CC5LR6 5679 IC50 > 500000 nM T04820 CNC40K 5680 IC50 > 500000 nM T04820 CKEB49 5681 IC50 > 500000 nM T04820 COC80L 85517 IC50 = 11000 nM T04820 CRP4A8 244537 IC50 = 5100 nM T04820 CWPG52 287041 IC50 = 16500 nM T04820 C84TRA 306203 IC50 = 600 nM T04820 C53ACF 306810 IC50 = 48400 nM T04820 CUDP24 449240 IC50 > 500000 nM T04820 CRO8F0 478671 IC50 = 4700 nM T04820 CAJ0G3 505777 IC50 = 130 nM T04820 C2ZVI7 505780 IC50 = 3500 nM T04820 C4DXN9 682361 IC50 = 4000 nM T04820 C69BXI 682362 IC50 = 4000 nM T04820 CZT9R1 698287 IC50 = 41700 nM T04820 CH6W9V 725903 IC50 > 37000 nM T04820 CR1WK8 765332 IC50 = 13100 nM T04820 C7JP0N 779201 IC50 = 69000 nM T04820 C24KUJ 837245 IC50 = 700 nM T04820 CS4WK1 947949 IC50 = 3500 nM T04820 CT78EF 954131 IC50 = 24000 nM T04820 C37JPW 1238707 IC50 = 17100 nM T04820 CCP95T 1240986 IC50 > 19000 nM T04820 C24MXJ 1379197 IC50 = 11000 nM T04820 CM0QX7 2047325 IC50 = 17000 nM T04820 C3IKV5 2774222 IC50 = 87000 nM T04820 CH6I4D 3517770 IC50 = 10000 nM T04820 C0M7EO 4058442 IC50 = 45400 nM T04820 C3FSL2 4626944 IC50 = 15900 nM T04820 CH37FE 5275722 IC50 = 14000 nM T04820 CX2O6U 5354063 IC50 = 22000 nM T04820 CI5MO8 5376379 IC50 = 20000 nM T04820 CR6LX3 5378133 IC50 = 268000 nM T04820 CZ5FA9 5378325 IC50 = 138000 nM T04820 CL41GY 5390853 IC50 = 3600 nM T04820 CTM1O5 5463500 IC50 > 256000 nM T04820 C0E6JW 5477132 IC50 = 3100 nM T04820 CST49O 5702960 IC50 = 17000 nM T04820 CI19NU 5708687 IC50 > 100000 nM T04820 CRE74N 5713385 IC50 > 37000 nM T04820 CT9Z7X 6476742 IC50 = 100000 nM T04820 CO68CR 6918711 IC50 = 1400 nM T04820 CZ9A7O 10023064 IC50 = 2500 nM T04820 C4RJ5M 10315303 IC50 = 2900 nM T04820 CF0B6P 11807517 IC50 = 29000 nM T04820 CQJE65 11989520 IC50 = 187000 nM T04820 C48HZD 12364579 IC50 = 38300 nM T04820 C2R9XW 12621903 IC50 < 371000 nM T04820 C09QFJ 13717983 IC50 = 182000 nM T04820 C13XHV 14069754 IC50 = 46200 nM T04820 CEA72J 14936055 IC50 > 44000 nM T04820 CXOR24 21822989 IC50 = 25000 nM T04820 CYD7W5 24426485 IC50 > 100000 nM T04820 CCS97Q 44329224 IC50 = 102000 nM T04820 CFQC08 44329248 IC50 = 539000 nM T04820 C5NOR7 44350539 IC50 > 21000 nM T04820 CI8EW1 44350563 IC50 = 2900 nM T04820 C3DG6P 44396811 IC50 = 26000 nM T04820 C52UQA 44396818 IC50 = 35000 nM T04820 CPYN39 44396824 IC50 = 61000 nM T04820 CQ60NW 44396859 IC50 = 35800 nM T04820 CI3V1Y 44396873 IC50 = 70000 nM T04820 C9TEU8 44419434 IC50 = 50000 nM T04820 CE5A4J 44591876 IC50 = 34000 nM T04820 CSW2X1 44591967 IC50 = 38000 nM T04820 C43NWV 44592001 IC50 = 61000 nM T04820 C7G0QO 49798419 IC50 = 600 nM T04820 CL1TN8 49798456 IC50 = 50200 nM T04820 C0WCG5 49798457 IC50 = 15100 nM T04820 CF35MO 49798508 IC50 = 700 nM T04820 C6QO2C 49798509 IC50 = 332800 nM T04820 C1D8NW 49798510 IC50 = 31500 nM T04820 CGE5L8 49798511 IC50 = 300 nM T04820 C8MP6E 49798512 IC50 = 29700 nM T04820 C65MWB 49798513 IC50 = 19700 nM T04820 CCMV23 49798553 IC50 = 127200 nM T04820 C7FQT0 49798554 IC50 = 20700 nM T04820 C0N1KX 49798555 IC50 = 40100 nM T04820 CKL1V8 49798556 IC50 = 600 nM T04820 C5K3NB 49798557 IC50 = 800 nM T04820 C5I2WJ 135906479 IC50 = 30000 nM T04820 CD70AY 135959419 IC50 > 57000 nM T04820 D00RIX 5280443 IC50 = 7000 nM T04820 D01SLS 4217 IC50 > 500000 nM T04820 D02NGU 3540 IC50 = 70000 nM T04820 D03OKV 9844320 IC50 > 10000 nM T04820 D04PTI 44591968 IC50 = 9000 nM T04820 D05SZP 5355577 IC50 = 17000 nM T04820 D06CTS 2735782 IC50 = 17400 nM T04820 D06WUE 49798484 IC50 = 600 nM T04820 D07OAT 456214 IC50 = 26000 nM T04820 D08FZK 44591969 IC50 = 18000 nM T04820 D09FFE 449241 IC50 > 500000 nM T04820 D0A6YW 5712235 IC50 = 8200 nM T04820 D0C8BV 3544 IC50 = 700 nM T04820 D0D8MA 15740307 IC50 = 200 nM T04820 D0E4AB 259098 IC50 = 400 nM T04820 D0F1KM 5784790 IC50 = 12000 nM T04820 D0G2DQ 4669250 IC50 = 5900 nM T04820 D0H3EV 5005498 IC50 = 51000 nM T04820 D0KH5T 5687 IC50 = 168000 nM T04820 D0Q3RF 44396914 IC50 = 18000 nM T04820 D0Q4PQ 5712110 IC50 = 10000 nM T04820 D0T3PW 5281672 IC50 = 157000 nM T04820 D0TO6S 2396 IC50 = 24000 nM T04820 D0UH0Q 6918599 IC50 = 18000 nM T04820 D0V5ZI 44419435 IC50 = 19000 nM T04820 D0V8JJ 5720587 IC50 = 1300 nM T04820 D0Y0ES 3707 IC50 = 30000 nM T04820 D0Y1UL 10561847 IC50 > 42000 nM T04820 D0Z6LR 29098931 IC50 = 14900 nM T78650 C0K6ZH 46934436 IC50 = 8000 nM T78650 C0DEA9 46934437 IC50 = 10000 nM T78650 C1SU7X 49864806 IC50 = 32000 nM T78650 C8WA3I 49864807 IC50 = 100000 nM T78650 CWPT38 49864808 IC50 = 60000 nM T78650 CDK39J 49864871 IC50 = 80000 nM T78650 CB7K5Z 49864872 IC50 = 35000 nM T78650 CSE5H0 49864873 IC50 = 85000 nM T78650 C4U2AX 49864909 IC50 = 32000 nM T78650 CPI7U5 49864910 IC50 = 60000 nM T78650 C03CNK 49864942 IC50 = 25000 nM T78650 CT98XD 49865001 IC50 = 60000 nM T78650 C3T0ZC 49865002 IC50 = 60000 nM T78650 C6ZKA1 49865003 IC50 = 150000 nM T78650 C3F4JS 49865004 IC50 = 80000 nM T93105 C5M2QY 2116 EC50 > 100000 nM T93105 CZN6S9 743974 EC50 > 25118.86 nM T93105 CDCS01 10206564 EC50 = 4000 nM T93105 C0QNE9 10435235 EC50 = 0.114 nM T93105 C4ESM9 20632905 EC50 > 100000 nM T93105 CTF47W 25164607 IC50 = 1.3 nM T93105 CTB5M4 25164609 IC50 = 5 nM T93105 CEKW51 25164812 IC50 = 6 nM T93105 C54DIT 25179907 EC50 = 11300 nM T93105 CM3H5J 46837918 EC50 = 4600 nM T93105 CY3OX0 53363314 EC50 = 1100 nM T93105 CWX1L8 58445338 IC50 = 18 nM T93105 C2BU7K 58445348 IC50 = 320 nM T93105 C8K7BT 71453301 IC50 = 8 nM T93105 CLC41Y 71458663 IC50 = 377 nM T93105 C61FYG 71460487 IC50 = 22 nM T93105 C5Y1GS 71462196 IC50 = 24 nM T93105 CVP73G 71682215 EC50 = 2000 nM T93105 C2CZ4D 71682359 IC50 = 39810.72 nM T93105 C18XRV 71682361 IC50 = 25118.86 nM T93105 C5IQJ3 71682362 EC50 = 10000 nM T93105 CN4B6I 71682363 EC50 = 9000 nM T93105 CBUW31 71682510 EC50 = 10000 nM T93105 CK63BG 71682511 EC50 = 8000 nM T93105 C9WVJ7 71682513 EC50 = 11000 nM T93105 C1A7PW 71682514 EC50 = 5000 nM T93105 C7AMD3 71682515 EC50 = 6000 nM T93105 C9IAV4 71682664 EC50 = 13000 nM T93105 C80EQR 71682665 EC50 = 1000 nM T93105 CT8P6A 73352089 EC50 = 6000 nM T93105 CTXA23 118726936 EC50 = 12000 nM T93105 C2FWY0 118726937 EC50 = 15600 nM T93105 C6XH0K 118726938 EC50 = 14100 nM T93105 CE7L6H 118726939 EC50 = 2500 nM T93105 CMN5S3 118726940 EC50 = 4400 nM T93105 C8LJ3F 118726941 EC50 = 3200 nM T93105 CD4A1T 118726942 EC50 = 1800 nM T93105 CB23OM 118726943 IC50 = 7000 nM T93105 CVU2B8 118726944 EC50 = 3200 nM T93105 C7EU9N 118726945 EC50 = 1000 nM T93105 CXEG20 118726946 EC50 = 23200 nM T93105 CMS2J7 118726947 EC50 = 2100 nM T93105 CHM38G 118726948 EC50 = 10700 nM T93105 CY3J0G 118726949 IC50 = 630 nM T93105 C94HSX 118726950 EC50 = 2200 nM T93105 CR6IC4 118726951 EC50 = 4500 nM T93105 C4J5EW 118726952 EC50 = 970 nM T93105 C8GOD6 118726953 EC50 > 40000 nM T93105 CVO6Y5 118726954 EC50 = 11200 nM T93105 CA8TS2 118726955 EC50 = 1100 nM T93105 C89LIX 118726956 EC50 = 1300 nM T77537 D09KTS 24821094 IC50 = 3 nM T77537 D0E6XR 3062316 IC50 = 228 nM T77537 D02NNV 3038525 IC50 > 10000 nM T77537 D02TUL 118115473 Ki = 26.9 nM T77537 D08AOZ 86582336 IC50 = 410 nM T77537 D0E3TC 44259 IC50 = 10 nM T77537 D0G5XV 135565884 IC50 = 56 nM T77537 D0LF1U 5287969 IC50 > 14850 nM T77537 D0S5RC 3025986 IC50 > 40000 nM T77537 D0YB3W 156414 IC50 = 5650 nM T77537 D03BNU 59604787 IC50 > 10000 nM T77537 D0LF0O 135441202 IC50 = 370 nM T77537 C9VW8M 449054 IC50 > 16000 nM T77537 CED2F1 668334 Ki = 460 nM T77537 CB6R5K 3722581 Ki = 15 nM T77537 CTID76 5282335 IC50 = 29000 nM T77537 CUCE63 5329663 IC50 > 10000 nM T77537 C8SU6K 9806812 IC50 = 1000 nM T77537 CM5Z8X 9869943 IC50 > 10000 nM T77537 CERH18 9871955 IC50 = 540 nM T77537 CV02OT 9914277 IC50 = 970 nM T77537 CQ2S4D 9964914 Ki = 3000 nM T77537 C7YD1X 10048045 IC50 > 25000 nM T77537 CXG4Q9 10110453 IC50 = 4800 nM T77537 CF34HN 10114123 IC50 = 950 nM T77537 CVM07F 10120124 IC50 = 230 nM T77537 C7R9GF 10151801 IC50 = 250 nM T77537 C28JIN 10151831 IC50 = 160 nM T77537 C1Q9PD 10152000 IC50 = 1100 nM T77537 CZ4JE8 10160476 IC50 = 92 nM T77537 CG1FZ5 10162990 IC50 = 270 nM T77537 C6QU7V 10163233 IC50 = 1300 nM T77537 C2G5HY 10165201 IC50 = 260 nM T77537 C9J2KW 10181704 IC50 = 690 nM T77537 CK0SX4 10194689 IC50 = 1600 nM T77537 C5PKO2 10195094 IC50 = 370 nM T77537 CD18OB 10195108 IC50 = 69 nM T77537 CXI97Z 10195393 IC50 = 7400 nM T77537 CF84LX 10195646 IC50 = 60 nM T77537 CGM5W0 10217158 IC50 = 390 nM T77537 CKH5C7 10217329 IC50 = 7200 nM T77537 C9R7FB 10224336 IC50 = 190 nM T77537 C2ODX6 10228329 IC50 = 76 nM T77537 CQ3Z6X 10230606 IC50 = 81 nM T77537 CSGD16 10246246 IC50 > 7000 nM T77537 C89JTD 10288201 IC50 = 330 nM T77537 CXS48F 10288395 IC50 = 110 nM T77537 C4QR0P 10301758 IC50 = 940 nM T77537 C47LSO 10310783 IC50 = 140 nM T77537 C5TYO0 10310880 IC50 = 730 nM T77537 CJ7U4I 11161778 IC50 = 17000 nM T77537 C2W5RC 11235063 IC50 > 50000 nM T77537 CRK56F 11237786 IC50 = 650 nM T77537 CBOP58 11293798 Ki > 10000 nM T77537 CJ8A6Y 11341428 IC50 = 820 nM T77537 C26BZX 11362471 Ki > 10000 nM T77537 CWXB93 11397177 Ki > 10000 nM T77537 CEP8N2 11489351 IC50 = 2 nM T77537 CRU9D3 11508262 Ki = 210 nM T77537 C4BK1O 11514905 Ki > 30000 nM T77537 CKX45I 11536964 Ki > 6000 nM T77537 CTG83F 11539329 Ki > 3800 nM T77537 CPW27V 11581044 Ki = 120 nM T77537 CMIL86 11590363 Ki > 3800 nM T77537 CJU5W6 11611103 Ki = 112 nM T77537 CI8CR3 11623444 Ki = 1300 nM T77537 C3UDF2 11623669 Ki = 1200 nM T77537 CK34LS 11632737 IC50 > 50000 nM T77537 C9T6SC 11640926 Ki > 3800 nM T77537 C5B6KR 11660004 Ki = 280 nM T77537 CLXI20 11675164 Ki = 220 nM T77537 CHSL63 11688314 Ki = 530 nM T77537 CU0E8O 11690457 Ki > 10000 nM T77537 CB16DG 11695198 Ki = 2100 nM T77537 CB0AP2 11705863 Ki > 10000 nM T77537 CE49IU 11718919 Ki > 2000 nM T77537 C45EWD 11723489 IC50 > 7000 nM T77537 CFPW41 16007116 Ki > 1500 nM T77537 CKR57M 16086104 IC50 > 5000 nM T77537 C16NRY 16086114 IC50 > 25000 nM T77537 CQG45C 16109001 IC50 = 25000 nM T77537 C1U8XW 16109036 IC50 > 5000 nM T77537 CGC34R 16118737 IC50 > 25000 nM T77537 C0H8UN 16730109 IC50 > 50000 nM T77537 CEW2T0 17501441 Ki > 4 nM T77537 CAF64K 20635205 IC50 = 30 nM T77537 CNLC10 20635235 IC50 = 7 nM T77537 C4PXQ6 20635236 IC50 = 6 nM T77537 C5LS4A 20635249 IC50 = 7 nM T77537 CD04JU 20635261 IC50 = 83 nM T77537 CPQ1F9 20635262 IC50 = 34 nM T77537 C3OH6S 20635263 IC50 = 15 nM T77537 C4XGT7 20635267 IC50 = 370 nM T77537 CTA9W2 20635268 IC50 = 320 nM T77537 CZ4W7A 20635392 IC50 = 2400 nM T77537 C16JNA 20635396 IC50 = 96 nM T77537 C3F4MT 20635404 IC50 = 40 nM T77537 C7NZ2P 20635405 IC50 = 35 nM T77537 C1ITS2 20635410 IC50 = 350 nM T77537 C75ATW 20635412 IC50 = 34 nM T77537 C4DAM0 20635501 IC50 = 250 nM T77537 C1V2MY 20635507 IC50 = 7 nM T77537 CB9E7N 20635510 IC50 = 19 nM T77537 C0XIQ2 20635514 IC50 = 12 nM T77537 COV49P 20635515 IC50 = 14 nM T77537 C2V5RM 20635525 IC50 = 18 nM T77537 CA12GX 20635526 IC50 = 29 nM T77537 CDTH82 20635527 IC50 = 47 nM T77537 CK2X6E 20635530 IC50 = 20 nM T77537 C8T7OA 20635534 IC50 = 9 nM T77537 CM83LK 20635537 IC50 = 260 nM T77537 CA61QF 21083895 IC50 = 9100 nM T77537 C6SL2R 22170396 IC50 = 60 nM T77537 C2FHR8 22170398 IC50 = 90 nM T77537 C0A8BN 22170403 IC50 = 290 nM T77537 CMNU25 22170411 IC50 = 930 nM T77537 CL9IA2 22170419 IC50 = 30 nM T77537 CRK8D4 22170436 IC50 = 210 nM T77537 CH5T9P 22170437 IC50 = 2190 nM T77537 C6JV7W 23400934 IC50 > 7000 nM T77537 CD5S7O 23401001 IC50 > 7000 nM T77537 CF67IQ 23628269 IC50 = 40 nM T77537 C7YG1N 24759534 IC50 = 26 nM T77537 CQNP54 24764449 IC50 = 62 nM T77537 C2UOE0 24766030 IC50 > 20000 nM T77537 CY8X0J 24811794 Ki > 10000 nM T77537 C9F1AO 24821023 IC50 = 11 nM T77537 CS3Q8B 24995659 IC50 > 2000 nM T77537 C0B7RT 25057409 IC50 > 10000 nM T77537 C0K9HA 25110600 IC50 = 46 nM T77537 CSNC57 25110758 IC50 = 3 nM T77537 C0GOX5 25110759 IC50 = 6 nM T77537 CC2R7S 25110760 IC50 = 7 nM T77537 CL82CU 25110796 IC50 = 4 nM T77537 CHT0B4 25169252 IC50 = 280 nM T77537 CJL25F 25169253 IC50 = 410 nM T77537 C2RX6E 25190503 IC50 = 3 nM T77537 CFN61D 25190504 IC50 = 170 nM T77537 C8LQS3 25190505 IC50 = 26 nM T77537 C20WQJ 25190506 IC50 > 5000 nM T77537 CM61RX 25190507 IC50 = 90 nM T77537 C5UCN3 25190508 IC50 = 2500 nM T77537 CTVK31 25190509 IC50 = 95 nM T77537 CY43QX 25190510 IC50 = 14 nM T77537 C09SGT 25190511 IC50 = 57 nM T77537 C9O0AL 25190512 IC50 = 340 nM T77537 C6RC2N 25190513 IC50 = 130 nM T77537 CA9U5F 25190514 IC50 = 450 nM T77537 C1ZCK4 25190515 IC50 = 170 nM T77537 CBX7Z3 25190516 IC50 = 180 nM T77537 CY3X8L 25190517 IC50 = 10 nM T77537 CONP02 25190518 IC50 = 14 nM T77537 CL81KR 25190519 IC50 = 100 nM T77537 C2I6JX 25190520 IC50 = 15 nM T77537 C8TK1S 25190521 IC50 = 2 nM T77537 CHD51B 25190522 IC50 = 14 nM T77537 C0G9EX 25190523 IC50 = 570 nM T77537 CUJS83 25190524 IC50 = 55 nM T77537 CE3W4R 25190525 IC50 = 140 nM T77537 CIAB51 25190526 IC50 = 1200 nM T77537 CA4Z2Y 25190527 IC50 = 5 nM T77537 C8OW9I 25190528 IC50 = 100 nM T77537 C5PH6D 25190529 IC50 = 740 nM T77537 CZ46JX 25190530 IC50 = 50 nM T77537 CE3T5U 25190531 IC50 = 6 nM T77537 CEHP95 25190532 IC50 = 190 nM T77537 C06LXS 25190533 IC50 = 10 nM T77537 C9RXL3 25190534 IC50 = 2 nM T77537 CC1E3O 25190535 IC50 = 13 nM T77537 C1NZ4D 25190536 IC50 = 81 nM T77537 CNR75T 25190537 IC50 = 380 nM T77537 C7LMI1 25190538 IC50 = 150 nM T77537 CLU7D2 25190539 IC50 = 74 nM T77537 CD2Z1T 25190540 IC50 = 8 nM T77537 CUP7E4 25190541 IC50 = 60 nM T77537 C57KGJ 25190542 IC50 = 10 nM T77537 CF9C5J 25190543 IC50 = 5 nM T77537 C3KJ6P 25190544 IC50 = 2 nM T77537 CU6VA8 25190545 IC50 = 7 nM T77537 CR0JP6 25190546 IC50 = 390 nM T77537 CJLB59 25190547 IC50 = 10 nM T77537 C27RCT 25190548 IC50 = 11 nM T77537 CM7A8T 25190549 IC50 = 6 nM T77537 C3YA7U 25190550 IC50 = 5 nM T77537 C6SE7Y 25190551 IC50 = 65 nM T77537 CPK7E0 25190552 IC50 = 67 nM T77537 CA2K4Q 25190553 IC50 = 13 nM T77537 CWRO62 25190554 IC50 = 58 nM T77537 C5UFS2 25190555 IC50 = 270 nM T77537 C6J2UZ 25190556 IC50 = 30 nM T77537 CMP9A2 25190557 IC50 = 130 nM T77537 CKP50F 25190558 IC50 = 6 nM T77537 CE3W9P 25190559 IC50 = 9 nM T77537 CNBO46 25190560 IC50 = 6 nM T77537 CCP4K9 25190561 IC50 = 42 nM T77537 CYK5Z2 25190562 IC50 = 740 nM T77537 C25JMO 25190563 IC50 = 8 nM T77537 CJ4W6E 25190564 IC50 = 12 nM T77537 CBV3D6 25190565 IC50 = 7 nM T77537 CE9UI6 25190566 IC50 = 37 nM T77537 CAK4E6 25190567 IC50 = 63 nM T77537 CTR6A2 25190568 IC50 = 39 nM T77537 CC40BJ 25190569 IC50 = 75 nM T77537 C7B6OS 25190570 IC50 = 39 nM T77537 CCJY98 25190571 IC50 = 59 nM T77537 C57PDK 25191024 IC50 = 510 nM T77537 CN5E0F 25263283 IC50 = 19000 nM T77537 CB8YN2 44201333 IC50 = 1 nM T77537 C8KNA3 44219632 Ki > 4000 nM T77537 C0VIX4 44219633 Ki > 4000 nM T77537 C39MDP 44410415 IC50 = 5000 nM T77537 CAMH81 44410416 IC50 = 14000 nM T77537 CW4U8D 44410417 IC50 = 4600 nM T77537 CEWY72 44410418 IC50 = 1700 nM T77537 CBZ9G1 44410419 IC50 = 730 nM T77537 CB16MX 44410420 IC50 = 2200 nM T77537 CM4J5W 44410421 IC50 = 2100 nM T77537 C5VR2O 44410424 IC50 = 2420 nM T77537 C32GPA 44410428 IC50 = 1090 nM T77537 C9E7KL 44410430 IC50 = 1030 nM T77537 CL7W3J 44410455 IC50 = 2600 nM T77537 CQLO41 44410456 IC50 = 900 nM T77537 CW7A2I 44410457 IC50 = 39000 nM T77537 C3HK5U 44410461 IC50 = 14800 nM T77537 C1Z3YU 44410513 IC50 > 50000 nM T77537 CQX90C 44410514 IC50 = 1600 nM T77537 CTFW82 44410519 IC50 = 1600 nM T77537 CN2A5F 44410567 IC50 = 600 nM T77537 C9M2AF 44410577 IC50 = 37000 nM T77537 C6SN3R 44410609 IC50 = 380 nM T77537 CKBT38 44410612 IC50 > 50000 nM T77537 C1FMC7 44410613 IC50 > 50000 nM T77537 C8QW6B 44410614 IC50 > 50000 nM T77537 CT6PH4 44410617 IC50 > 50000 nM T77537 CW93VP 44410622 IC50 = 13000 nM T77537 CFQ6I2 44410627 IC50 = 1440 nM T77537 CDB3X8 44410652 IC50 = 260 nM T77537 C6ZMA0 44410656 IC50 = 15000 nM T77537 C1FR5B 44410659 IC50 > 50000 nM T77537 CGA70U 44410660 IC50 > 50000 nM T77537 CB32UG 44410662 IC50 > 50000 nM T77537 C6E0TJ 44410667 IC50 > 50000 nM T77537 CR9LC6 44410668 IC50 = 11200 nM T77537 CARJ28 44410676 IC50 = 5700 nM T77537 CT9G0X 44410737 IC50 = 350 nM T77537 CLVC63 44410741 IC50 = 720 nM T77537 CA7ZC5 44410746 IC50 = 2000 nM T77537 CKI8M1 44412537 IC50 = 600 nM T77537 C8LDU0 44412550 IC50 = 820 nM T77537 C1Y7OA 44412551 IC50 = 3900 nM T77537 CTM8Z6 44412588 IC50 = 22340 nM T77537 CRG1L6 44412606 IC50 > 25000 nM T77537 C4NUK8 44412771 IC50 = 1130 nM T77537 CC0WJ8 44412792 IC50 = 19240 nM T77537 C5G4SU 44413075 IC50 > 50000 nM T77537 CADR04 44413087 IC50 = 46300 nM T77537 CG8NE2 44413088 IC50 = 6060 nM T77537 C7OF0Q 44413100 IC50 = 7070 nM T77537 COH5J0 44413186 IC50 = 34200 nM T77537 CMVT21 44432424 IC50 = 2700 nM T77537 CPX6K4 44432425 IC50 = 62 nM T77537 C6A3NK 44432426 IC50 > 20000 nM T77537 CD4Q5O 44432427 IC50 > 20000 nM T77537 CI95MW 44432428 IC50 > 20000 nM T77537 CJ1FH3 44432429 IC50 = 11000 nM T77537 CW5J2A 44432432 IC50 = 20000 nM T77537 CU90YD 44432433 IC50 = 12000 nM T77537 CA38PO 44432438 IC50 = 11000 nM T77537 CH4DL7 44432439 IC50 > 20000 nM T77537 C46ZFU 44432440 IC50 = 1700 nM T77537 CA98KR 44432441 IC50 = 110 nM T77537 C3VRO9 44557921 IC50 > 10000 nM T77537 CJAV21 44573146 IC50 = 3 nM T77537 CP9E4J 44573266 IC50 = 100 nM T77537 CLA24D 44573267 IC50 = 11 nM T77537 C51CDF 44573268 IC50 = 8 nM T77537 CDT4K9 44573269 IC50 = 940 nM T77537 CD8Q5P 44573306 IC50 = 780 nM T77537 C5CA0V 44573307 IC50 = 2 nM T77537 CNMO98 44573308 IC50 = 2 nM T77537 CAZ59C 44573309 IC50 = 20 nM T77537 C7T3HJ 44573374 IC50 = 4 nM T77537 CPMG47 44573375 IC50 = 2 nM T77537 CT1R3Z 44573376 IC50 = 3 nM T77537 CF3N7G 44573377 IC50 = 140 nM T77537 C6BRV7 44573424 IC50 = 1 nM T77537 CXU7T6 44573425 IC50 = 2 nM T77537 C81CVB 44573426 IC50 = 1 nM T77537 CS27CU 44573427 IC50 = 3 nM T77537 CAYJ73 44573467 IC50 = 1 nM T77537 CN6G1U 44573468 IC50 = 8 nM T77537 CO4N5B 44573469 IC50 = 2 nM T77537 CDU34Y 44573502 IC50 = 3 nM T77537 CY81WI 44573503 IC50 = 660 nM T77537 CM9E7S 44573504 IC50 = 2 nM T77537 C42NEB 44573505 IC50 = 1 nM T77537 CK24OS 44573546 IC50 = 2 nM T77537 C53MYT 44588579 IC50 = 10 nM T77537 CSY05L 44588580 IC50 = 27 nM T77537 CSV19C 44588581 IC50 = 18 nM T77537 CKN87Z 44588582 IC50 = 46 nM T77537 CJB84Y 44588583 IC50 = 8 nM T77537 CI30GZ 44588584 IC50 = 76 nM T77537 C2C6XI 44588606 IC50 = 54 nM T77537 CU4A2I 44588607 IC50 = 3 nM T77537 C6Z3CL 44588719 IC50 = 10 nM T77537 CXN8P2 44588738 IC50 = 5 nM T77537 CNPI73 44588739 IC50 = 10 nM T77537 CK34PA 44588740 IC50 = 25 nM T77537 CL67AQ 44588741 IC50 = 16 nM T77537 C6JVC8 44588765 IC50 = 9 nM T77537 C0C9UI 44588766 IC50 = 3 nM T77537 CT6VG5 44588767 IC50 = 10 nM T77537 CZ1P6B 44588791 IC50 = 12 nM T77537 CWJ92G 44588792 IC50 = 3300 nM T77537 C4U8BY 44588793 IC50 = 56 nM T77537 CU6O3G 44588794 IC50 = 35 nM T77537 C30HRN 44588845 IC50 = 4 nM T77537 CY5T8I 44588846 IC50 = 68 nM T77537 C1YI7Z 44588847 IC50 = 250 nM T77537 CK79TL 44588878 IC50 = 4500 nM T77537 CML1U9 44588879 IC50 = 520 nM T77537 C10BIC 44588880 IC50 > 10000 nM T77537 C3JS6Q 44588881 IC50 = 270 nM T77537 C2VDN8 44588915 IC50 = 16 nM T77537 CSC84A 44588916 IC50 = 4500 nM T77537 C4FIC7 44588917 IC50 = 35 nM T77537 C4Z1DQ 44588918 IC50 = 6 nM T77537 CKB0C7 44588945 IC50 = 89 nM T77537 CG6RP1 44588946 IC50 = 690 nM T77537 CJ6BN1 44588947 IC50 = 2000 nM T77537 CLO50G 44588965 IC50 = 2 nM T77537 CLA8G9 44588966 IC50 = 12 nM T77537 CV03WM 44588967 IC50 = 16 nM T77537 C5I7DE 44588968 IC50 = 73 nM T77537 C82SKN 44588969 IC50 = 9 nM T77537 CTL5U3 44588970 IC50 = 14 nM T77537 CFYP17 44588994 IC50 = 10 nM T77537 CRU7I3 44588995 IC50 = 1100 nM T77537 CQR2N6 44588996 IC50 = 35 nM T77537 C3J7WS 44588997 IC50 = 4 nM T77537 C0UFA7 44588998 IC50 = 61 nM T77537 C4S3ZD 44588999 IC50 = 5 nM T77537 CUY54I 44589015 IC50 = 27 nM T77537 C5RG0W 44589016 IC50 = 1900 nM T77537 C6QFD0 44589017 IC50 = 5 nM T77537 CW2DV3 44589018 IC50 = 18 nM T77537 CEGF45 44589019 IC50 > 20000 nM T77537 CWO6V3 44589020 IC50 > 20000 nM T77537 C6FJ7Y 44589021 IC50 = 7 nM T77537 CXE42M 44589045 IC50 = 23 nM T77537 CC4DW7 44589046 IC50 = 150 nM T77537 CCJM31 44589047 IC50 = 59 nM T77537 C7NRT2 44589048 IC50 = 320 nM T77537 CATZ92 44589049 IC50 = 220 nM T77537 CG1X2R 44589639 IC50 = 170 nM T77537 C7Y2UR 44589640 IC50 = 45 nM T77537 CKU74A 44589641 IC50 = 48 nM T77537 CB06FP 44589642 IC50 = 34 nM T77537 CH4OB9 44589677 IC50 = 81 nM T77537 CU3MJ6 44589678 IC50 = 69 nM T77537 CYDZ59 44589679 IC50 > 10000 nM T77537 CDJ51R 44589680 IC50 = 46 nM T77537 CNI87X 44589716 IC50 = 20 nM T77537 CEZ4C6 44589717 IC50 = 1200 nM T77537 CJ8P0D 44589718 IC50 = 47 nM T77537 CKE0R1 44589719 IC50 = 36 nM T77537 CT3W7G 44589754 IC50 = 6 nM T77537 C7PMB4 44589755 IC50 = 41 nM T77537 CLI17Q 44589756 IC50 = 30 nM T77537 C9MDA8 44589757 IC50 = 27 nM T77537 CK2L6P 44589793 IC50 = 46 nM T77537 CY7HW6 44589794 IC50 = 53 nM T77537 CBW27Y 44589795 IC50 = 3 nM T77537 CO21BJ 44589832 IC50 = 110 nM T77537 CZL1U2 44593710 IC50 = 8 nM T77537 C9B7LK 44593713 IC50 = 4 nM T77537 CY3HW5 46224684 IC50 > 10000 nM T77537 C7H4YM 46865419 IC50 > 10000 nM T77537 CLS29B 46872626 IC50 > 10000 nM T77537 C2O8RZ 46886323 IC50 > 1000 nM T77537 C28ELR 46912278 Ki = 1.585 nM T77537 CD4L7V 46912279 Ki = 0.2512 nM T77537 C7S2HO 46913757 Ki = 0.1995 nM T77537 CT46HI 46913758 Ki = 0.2512 nM T77537 C9L3XR 49838879 IC50 > 50000 nM T77537 C5V9BE 52936431 Ki = 140 nM T77537 CR3X8W 52936432 Ki > 30000 nM T77537 C13LER 52936433 Ki = 170 nM T77537 C1VML8 52936434 Ki = 93 nM T77537 CU1T5C 52936530 Ki = 7 nM T77537 CK69ML 52936531 Ki = 16 nM T77537 CCT6B9 52936532 Ki = 46 nM T77537 CC7SE4 52936533 Ki = 145 nM T77537 CA93FM 52936534 Ki = 11 nM T77537 C9KO7D 52936535 Ki = 23 nM T77537 CEQN27 52936621 Ki = 7 nM T77537 C2A6MX 52936622 Ki = 20 nM T77537 CBH0K9 52936623 Ki = 20 nM T77537 CKF2D5 52936624 Ki = 27 nM T77537 CD4H3S 53354074 Ki > 1000 nM T77537 C8ZRE3 53356518 IC50 = 52 nM T77537 CN9QD7 56643097 IC50 > 10000 nM T77537 CJBL48 56925034 IC50 = 39 nM T77537 C7RDQ8 56925241 IC50 = 5 nM T77537 CT3EW2 59292007 IC50 > 1000 nM T77537 CZ3TG1 59375154 IC50 = 55 nM T77537 CXJ63M 59603829 IC50 = 94 nM T77537 CQEU96 59603842 IC50 = 26 nM T77537 CV63UL 67240318 IC50 > 10000 nM T77537 C5DGR9 69036886 IC50 = 10000 nM T77537 C3GTU1 69762142 IC50 > 10000 nM T77537 C7VJ6A 70647728 IC50 = 96 nM T77537 C5HB9I 71259491 Ki = 0.1 nM T77537 C6D0JX 71259500 Ki = 1.4 nM T77537 CP5O3N 71259506 Ki = 59 nM T77537 C64KQW 71259516 Ki = 6.6 nM T77537 CS92ID 71259555 Ki = 0.93 nM T77537 C2WL5D 71259557 Ki = 44 nM T77537 C7BNF0 71259563 Ki = 27 nM T77537 C4SJ1M 71259597 Ki = 7.8 nM T77537 CC96VO 71259598 Ki = 0.56 nM T77537 CK9MW3 71259641 Ki = 1 nM T77537 C4SPA0 71259651 Ki = 35 nM T77537 CJ4BK2 71259773 Ki = 10 nM T77537 CKH6Z3 71259783 Ki = 580 nM T77537 C1IZT4 71259797 Ki = 36 nM T77537 C9AF8W 71267243 Ki = 0.8 nM T77537 CE5SB7 71267246 Ki = 381 nM T77537 CG7U6V 71267305 Ki = 11 nM T77537 CI0R3A 71267318 Ki = 0.8 nM T77537 C5X2UZ 71267326 Ki = 0.23 nM T77537 C76CXB 71450143 IC50 = 2450 nM T77537 CY8X9L 71450144 IC50 > 100000 nM T77537 C4MBT3 71450145 IC50 = 720 nM T77537 C5YX9S 71450146 IC50 = 2 nM T77537 CYP5D9 71450147 IC50 = 6470 nM T77537 C2PV9H 71450148 IC50 = 1750 nM T77537 C9ID7H 71450149 IC50 = 780 nM T77537 CDLK74 71450150 IC50 = 65000 nM T77537 CA03KS 71450151 IC50 = 21417 nM T77537 CBMZ60 71450184 IC50 = 7457 nM T77537 CCYE35 71450185 IC50 = 4425 nM T77537 C34TYA 71450186 IC50 = 2495 nM T77537 C34MPQ 71451977 IC50 > 100000 nM T77537 CUK4C0 71451978 IC50 = 53650 nM T77537 C1CH6E 71451979 IC50 = 190 nM T77537 CWF2H0 71451980 IC50 = 180 nM T77537 CZL5M2 71451981 IC50 = 210 nM T77537 C0G3FM 71451982 IC50 > 100000 nM T77537 CQR24F 71453784 IC50 = 100 nM T77537 C8BLW0 71453785 IC50 = 10 nM T77537 CPA8Q9 71453786 IC50 = 520 nM T77537 CHM1S9 71453787 IC50 = 1520 nM T77537 CY0C7F 71453788 IC50 = 10880 nM T77537 C94XDU 71453789 IC50 = 36220 nM T77537 CNFQ61 71453790 IC50 > 100000 nM T77537 C3MYB5 71453818 IC50 = 52458 nM T77537 C49LMP 71455519 IC50 = 2180 nM T77537 C2R0KW 71455520 IC50 = 720 nM T77537 C7SX5M 71455521 IC50 = 1410 nM T77537 C6LH8Q 71455522 IC50 = 160 nM T77537 CL9YX8 71455523 IC50 = 10 nM T77537 C5B3VZ 71455524 IC50 > 100000 nM T77537 C9OZ7L 71455525 IC50 = 10324 nM T77537 CZE97Y 71455526 IC50 = 10068 nM T77537 CKT60L 71455860 Ki > 1500 nM T77537 C97EFZ 71457310 IC50 > 100000 nM T77537 C3ERY4 71457311 IC50 > 100000 nM T77537 CQBX94 71457312 IC50 = 130 nM T77537 CYIV59 71457313 IC50 = 4080 nM T77537 CM4XP7 71457314 IC50 > 100000 nM T77537 C7Y3CN 71457315 IC50 = 8341 nM T77537 CX9JD6 71457316 IC50 = 1045 nM T77537 COR7P9 71457317 IC50 = 22930 nM T77537 C6S2WH 71457340 IC50 = 21883 nM T77537 CNK30S 71459144 IC50 = 40 nM T77537 C2CMI9 71459145 IC50 = 5960 nM T77537 C7C5KR 71459146 IC50 = 73 nM T77537 CU6B3A 71459147 IC50 > 100000 nM T77537 CLN0C3 71459148 IC50 = 200 nM T77537 CS6JI3 71459149 IC50 = 1020 nM T77537 CKE8H3 71459150 IC50 = 2460 nM T77537 C4MA8X 71459191 IC50 = 20439 nM T77537 CLY18M 71460955 IC50 = 200 nM T77537 CQP21A 71460956 IC50 = 7570 nM T77537 CS3AW9 71460957 IC50 = 6645 nM T77537 C4LHT7 71462672 IC50 > 100000 nM T77537 CWD7E2 71462673 IC50 = 70 nM T77537 CX5K8Z 71462674 IC50 > 100000 nM T77537 C9FCM5 71462675 IC50 > 100000 nM T77537 CMF79G 71462676 IC50 = 21321 nM T77537 C8CG6H 71462712 IC50 = 9827 nM T77537 CEM84S 71462713 IC50 = 17744 nM T77537 CZM1K4 71765510 IC50 = 320 nM T77537 C98LKV 71777716 Ki = 8.4 nM T77537 C3MI4O 71777717 Ki = 0.7 nM T77537 C54XWG 72190869 IC50 > 10000 nM T77537 CS10DX 72544168 Ki = 1.9 nM T77537 CQH45K 72544389 Ki = 0.5 nM T77537 CVL5U1 72544390 Ki = 380 nM T77537 C2NV5Y 72544391 Ki = 2000 nM T77537 C21WYT 72544392 Ki = 230 nM T77537 CNOY69 72544393 Ki = 3500 nM T77537 CG38JZ 72544394 Ki = 50 nM T77537 CB9L0H 72544615 Ki = 85 nM T77537 C4OHT5 72544616 Ki = 3500 nM T77537 CA7C3K 72544617 Ki = 5.3 nM T77537 CJZV57 72544618 Ki = 6.6 nM T77537 CMS5O0 72544619 Ki = 2.5 nM T77537 CP7W1C 72544839 Ki = 30 nM T77537 CIE0T7 72544840 Ki = 1100 nM T77537 C0G4SO 72545063 Ki = 43 nM T77537 CFTK59 72705466 Ki > 10000 nM T77537 C1CU0H 72705467 Ki = 794.33 nM T77537 CX2AW3 72705468 Ki = 6.31 nM T77537 CVK4Z3 72705469 Ki = 501.19 nM T77537 C4ND6R 72705470 Ki = 63.1 nM T77537 CT67YO 72706106 Ki = 15.85 nM T77537 C9OQ2I 72710839 IC50 > 10000 nM T77537 C3L2WD 73292576 Ki = 5.3 nM T77537 C0P9LY 73292578 Ki = 10 nM T77537 CJ87SO 73292579 Ki = 75 nM T77537 CAS80Y 73292746 Ki = 8 nM T77537 C35BCQ 73292749 Ki = 37 nM T77537 C52LFH 73292907 Ki = 3 nM T77537 C0NE4O 73293422 Ki = 180 nM T77537 C26IVZ 73293424 Ki = 860 nM T77537 CIP49J 73293781 Ki < 0.1 nM T77537 CZ63BH 73293963 Ki = 42 nM T77537 CE1JT9 73294162 Ki = 0.3 nM T77537 C4FY5U 73346554 Ki = 0.3162 nM T77537 CPGD07 73348027 Ki = 3981.07 nM T77537 C05XEV 73348028 Ki = 158.49 nM T77537 CUW70Y 73348034 Ki = 0.3981 nM T77537 CFEU95 73348035 Ki = 15.85 nM T77537 C6K0UL 73348036 Ki > 10000 nM T77537 CD6KE7 73349574 Ki = 1.995 nM T77537 CV8UR4 73351136 Ki = 12.59 nM T77537 CAS60G 73352600 Ki = 3.981 nM T77537 CX75YR 73352604 Ki = 0.631 nM T77537 C5YKB4 73352605 Ki = 6.31 nM T77537 C03YUP 73355623 Ki = 19.95 nM T77537 C1A9PR 73357167 Ki = 1 nM T77537 CMEV76 74983355 Ki = 0.7 nM T77537 C0RP9Y 76309810 Ki = 0.6 nM T77537 C2A7SL 76320747 Ki = 6.4 nM T77537 CN39OQ 78341183 IC50 = 220 nM T77537 C1HW4B 89735655 IC50 = 4200 nM T77537 C5Q7UO 90036498 Ki = 31 nM T77537 C2ADJ1 90036634 Ki = 4000 nM T77537 CC06YJ 90036766 Ki = 22 nM T77537 CO51HL 90037453 Ki = 180 nM T77537 CX4C7W 90037556 Ki = 69 nM T77537 C6WQU2 90645540 Ki = 8.3 nM T77537 CSD73E 90645541 Ki = 0.8 nM T77537 C02KJP 90645542 Ki = 1.2 nM T77537 CE3OV2 90645543 Ki = 6.2 nM T77537 CY6L4N 90645544 Ki = 0.7 nM T77537 C7D5PI 90645545 Ki = 15 nM T77537 C93BGJ 90645546 Ki = 0.2 nM T77537 CSYV34 90656736 Ki = 3.4 nM T77537 C1CD8K 90656737 Ki = 1.7 nM T77537 C7C4KF 90656738 Ki > 4 nM T77537 CC6F3W 90656739 Ki = 53 nM T77537 CF89DA 90664659 IC50 = 22600 nM T77537 C64SIO 92042864 IC50 = 1070 nM T77537 C8HYU9 117926195 IC50 > 10000 nM T77537 CH4FU2 118641920 Ki = 0.27 nM T77537 C5EFI8 118641944 Ki = 14 nM T77537 CQ7Z0C 118641957 Ki = 8 nM T77537 CTP2E8 118737132 Ki = 0.5 nM T77537 C5GTM2 118737133 Ki = 0.2 nM T77537 C7MJ5H 118737134 Ki = 0.3 nM T77537 C3XF2A 118737135 Ki = 0.3 nM T77537 CNP5K8 118737136 Ki = 0.2 nM T77537 C8FDR1 118737137 Ki = 0.5 nM T77537 C37DUM 121293882 IC50 = 88 nM T77537 CXQR89 121294143 IC50 = 8.3 nM T77537 CFKD32 122191637 IC50 = 115 nM T77537 CLM7K3 122604539 IC50 > 10000 nM T77537 C01JHI 122604566 IC50 > 10000 nM T77537 CV89JM 132231876 IC50 = 23 nM T77537 C59HOQ 134277578 IC50 = 3.23 nM T77537 C0PZ5R 134277599 IC50 = 1.52 nM T77537 C7PWJ2 134277617 IC50 = 0.53 nM T77537 CRA2H1 134277633 IC50 = 1.5 nM T77537 CXJ8I0 134277643 IC50 = 0.34 nM T77537 C02RIA 134277647 IC50 = 0.67 nM T77537 CGH42R 134277652 IC50 = 0.72 nM T77537 COA14U 134277654 IC50 = 0.41 nM T77537 CQK0B5 134277685 IC50 = 10.1 nM T77537 C6S8VC 134277696 IC50 = 0.64 nM T77537 C49PIO 134277748 IC50 = 0.87 nM T77537 CD7VK4 134277767 IC50 = 1.62 nM T77537 CZ5E6L 134277773 IC50 = 0.7 nM T77537 C2CFK7 134277780 IC50 = 2.17 nM T77537 C6E7LW 134277790 IC50 = 0.81 nM T77537 C6T7NW 134277796 IC50 = 0.92 nM T77537 CU8ZP5 134277800 IC50 = 0.99 nM T77537 CTR4K6 134277828 IC50 = 0.58 nM T77537 C54FXD 134957362 IC50 > 10000 nM T77537 C6OE3V 135406885 IC50 = 160 nM T77537 COVY35 135406895 IC50 = 80 nM T77537 CUWM59 135409238 IC50 = 140 nM T77537 CG7K8I 135409247 IC50 = 170 nM T77537 CS0LR6 135445358 IC50 = 3980 nM T77537 CWM9Q1 135494486 IC50 = 350 nM T77537 C2U3AP 135514562 IC50 = 110 nM T77537 CK0M8W 135537103 IC50 = 250 nM T77537 CJ03PU 135566610 IC50 = 10.9 nM T77537 CQ9A5I 135566611 IC50 = 7 nM T77537 C42TOW 135566612 IC50 = 0.3 nM T77537 CN48IF 135566613 IC50 = 8.6 nM T77537 CIS2L5 135566617 IC50 = 150 nM T77537 C67IYS 135566618 IC50 = 1.9 nM T77537 CF48JM 135908497 IC50 = 560 nM T77537 C6H0AI 135957039 IC50 = 330 nM T77537 CP5SD0 136016241 IC50 = 2.4 nM T77537 CWB21F 136016374 IC50 = 2510 nM T77537 CCMG78 136016383 IC50 = 2000 nM T77537 CFTI43 136016384 IC50 = 1100 nM T77537 CBS87V 136016385 IC50 = 790 nM T77537 C05IWG 136016386 IC50 = 630 nM T77537 COPL16 136016393 IC50 = 630 nM T77537 C23APW 136016394 IC50 = 3160 nM T77537 C0XM8L 136016395 IC50 = 10000 nM T77537 CDS3A7 136016400 IC50 = 4360 nM T77537 CI37ET 136016401 IC50 = 1260 nM T77537 CD65WY 136016402 IC50 = 3160 nM T77537 CKWD23 136016403 IC50 = 1820 nM T77537 CO4C8Y 136016408 IC50 = 850 nM T77537 CUP47N 136016409 IC50 = 630 nM T77537 C4RMV8 136016410 IC50 = 1000 nM T77537 C0B7XQ 136016415 IC50 = 2060 nM T77537 C3Z6NG 136016416 IC50 = 1630 nM T77537 CXLZ12 136016417 IC50 = 2040 nM T77537 C9WVQ8 136016418 IC50 = 20400 nM T77537 C0MAS6 136016419 IC50 > 100000 nM T77537 C9BOX7 136016420 IC50 > 100000 nM T77537 C80OVA 136016421 IC50 = 630 nM T77537 C36PIS 136016422 IC50 = 500 nM T77537 CB8MI3 136016423 IC50 = 5000 nM T77537 CMY2N7 136016424 IC50 = 50100 nM T77537 CFY17E 136016425 IC50 = 1580 nM T77537 C7A9LY 136030592 IC50 = 120 nM T77537 CRA1H3 136030593 IC50 = 65 nM T77537 C4KLZ5 136030594 IC50 = 87 nM T77537 CVQF95 136030595 IC50 = 43 nM T77537 CRY2E5 136030598 IC50 = 140 nM T77537 CVZ3A4 136030599 IC50 = 260 nM T77537 C12OBR 136030600 IC50 = 70 nM T77537 C0Z7IM 136030629 IC50 = 20 nM T77537 CHMU19 136030633 IC50 = 110 nM T77537 CYRI63 136030634 IC50 = 100 nM T77537 CN3LU6 136030635 IC50 > 50000 nM T77537 C74LHJ 136030636 IC50 = 46 nM T77537 CFYO35 136030639 IC50 = 310 nM T77537 CP69FN 136030672 IC50 = 220 nM T77537 C6RIT2 136030673 IC50 > 50000 nM T77537 CF6D9C 136030674 IC50 = 66 nM T77537 CIC29X 136030675 IC50 = 120 nM T77537 CRY68L 136030705 IC50 = 190 nM T77537 C6Y0WA 136030710 IC50 = 370 nM T77537 CO4Z5H 136030736 IC50 = 67 nM T77537 C4S9QE 136030737 IC50 = 830 nM T77537 CPDZ24 136030738 IC50 = 45 nM T77537 C7GP4F 136030739 IC50 = 26 nM T77537 CLZ75U 136030740 IC50 = 85 nM T77537 CSA54K 136030741 IC50 = 730 nM T77537 C0TM4I 136030742 IC50 = 720 nM T77537 C4M9XD 136030743 IC50 = 10 nM T77537 CE9C0X 136030745 IC50 = 310 nM T77537 C1Z6KE 136030748 IC50 = 1500 nM T77537 C4U1ZE 136032568 IC50 = 240 nM T77537 CT3S7N 136032569 IC50 = 230 nM T77537 CO7BC1 136032578 IC50 = 22000 nM T77537 C5JM9H 136032600 IC50 = 80 nM T77537 C2JLY1 136032615 IC50 = 130 nM T77537 C0R9GU 136032627 IC50 = 90 nM T77537 CLR7S3 136059157 IC50 = 80 nM T77537 CUZ57E 136141542 IC50 = 2300 nM T77537 C9AT1U 136141543 IC50 = 98 nM T77537 CB74DR 136141544 IC50 = 900 nM T77537 C9PUM3 136141545 IC50 = 1410 nM T77537 C5YST1 136141546 IC50 = 750 nM T77537 CT6O7A 136141547 IC50 = 27 nM T77537 C71XIR 136141548 IC50 = 70 nM T77537 CK72XC 136141549 IC50 = 20 nM T77537 CS57KT 136141573 IC50 = 350 nM T77537 CNV86P 136141577 IC50 = 160 nM T77537 C5OW3D 136141585 IC50 = 530 nM T77537 C2AYS7 136141586 IC50 = 1000 nM T77537 C4C7OX 136141587 IC50 = 47 nM T77537 CYI26Q 136141588 IC50 = 72 nM T77537 C17KYN 136141589 IC50 = 1700 nM T77537 CY71KM 136141591 IC50 = 70 nM T77537 C7T0DC 136141592 IC50 = 1000 nM T77537 CLS79W 136141593 IC50 = 280 nM T77537 CZ7EX0 136183413 IC50 = 60 nM T77537 CQED29 136188798 IC50 = 140 nM T77537 CP5NE8 136188799 IC50 = 1600 nM T77537 CSRL54 136188800 IC50 = 36 nM T77537 C7VX4D 136188801 IC50 = 69 nM T77537 C9JS3P 136188802 IC50 = 250 nM T77537 CZ8IE1 136188803 IC50 = 340 nM T77537 CYLS64 136188804 IC50 = 300 nM T77537 CUE5X3 136188805 IC50 = 500 nM T77537 CU6Z0T 136188806 IC50 = 310 nM T77537 CJHT74 136188807 IC50 = 200 nM T77537 CTOR91 136188808 IC50 = 60 nM T77537 C9UIO6 136188809 IC50 = 110 nM T77537 CUI67Z 136188810 IC50 = 690 nM T77537 CUHP14 136188811 IC50 = 210 nM T77537 C9YLZ6 136188812 IC50 = 83 nM T77537 CPC8D4 136188813 IC50 = 780 nM T77537 C7TVJ9 136188814 IC50 = 860 nM T77537 C4AZP2 136188815 IC50 = 620 nM T77537 CI5V3P 136188816 IC50 = 1200 nM T77537 C28NFU 136188817 IC50 = 12000 nM T77537 C0BFO4 136188818 IC50 = 530 nM T77537 CB3IN0 136188819 IC50 = 16 nM T77537 CT9LV6 136188820 IC50 = 23 nM T77537 CD15JP 136188821 IC50 = 100 nM T77537 C9DU3V 136188822 IC50 = 100 nM T77537 CYZ9F4 136188823 IC50 = 990 nM T77537 CQL41E 136188824 IC50 = 260 nM T77537 CSH9W0 136188825 IC50 = 30 nM T77537 C1VJO0 136188826 IC50 = 77 nM T77537 C3UP6I 136188827 IC50 = 60 nM T77537 CW3E2V 136188828 IC50 = 130 nM T77537 CW1IV2 136199382 IC50 = 120 nM T77537 CJ0FZ4 136199383 IC50 = 190 nM T77537 CE27WO 136199384 IC50 = 80 nM T77537 C5Q0ZC 136199385 IC50 = 310 nM T77537 CB58FG 136199386 IC50 = 140 nM T77537 CTY4Q1 136199387 IC50 = 70 nM T77537 CY4TS0 136199388 IC50 = 200 nM T77537 C8EC0L 136199389 IC50 = 280 nM T77537 CSKP13 136199390 IC50 = 27000 nM T77537 CU8P2N 136199391 IC50 = 300 nM T77537 CRHS39 136199392 IC50 = 70 nM T77537 C26NEM 136254164 IC50 = 200 nM T77537 CXC69T 137321158 IC50 = 60 nM T77537 C3Z4AT 137321159 IC50 > 10000 nM T77537 C7TG3J 137641313 IC50 > 19952.62 nM T77537 C4DRX1 137643187 IC50 = 2190 nM T77537 C28QUP 137652864 IC50 = 5655 nM T77537 CRWA29 139030520 IC50 = 306.9 nM T77537 C9ZYG8 141366083 IC50 = 290 nM T77537 C4OD9Q 145967187 IC50 = 15.1 nM T77537 CE31VG 145979714 IC50 > 10000 nM T77537 C9BX4U 145988956 IC50 > 10000 nM T77537 C2MD1Q 155513187 IC50 > 10000 nM T77537 CA7O4B 155513491 IC50 = 5.4 nM T77537 C7AMX8 155514903 IC50 = 3.6 nM T77537 CI23DH 155516489 IC50 = 3.7 nM T77537 CU0VL1 155517584 IC50 = 22 nM T77537 C3NA2I 155519537 IC50 > 1000 nM T77537 CRT67D 155526236 IC50 = 1.3 nM T77537 CRC38Y 155526544 IC50 = 87 nM T77537 CE3OH1 155527121 IC50 < 1.26 nM T77537 CUXA18 155529935 IC50 = 2.3 nM T77537 CL0US4 155530459 IC50 = 0.5 nM T77537 C2WCU6 155530774 IC50 = 5.4 nM T77537 C1NGV5 155534208 IC50 = 3.7 nM T77537 C1UJ4T 155534213 IC50 = 32 nM T77537 CU9S7B 155535315 IC50 = 4.8 nM T77537 CBZ4V6 155536645 IC50 = 1437 nM T77537 C2CG1A 155537016 IC50 > 10000 nM T77537 C0JL6C 155537712 IC50 = 23 nM T77537 CWY1O0 155538122 IC50 > 10000 nM T77537 CJ5OI0 155541008 IC50 = 423 nM T77537 CH10DU 155542091 IC50 = 5.1 nM T77537 CELG50 155543350 IC50 = 469 nM T77537 CW73EO 155543439 IC50 < 1.26 nM T77537 CO1S0E 155546265 IC50 = 42 nM T77537 C2ZHA0 155547912 IC50 = 22 nM T77537 C0C1FI 155548702 IC50 = 126 nM T77537 C79PYG 155550586 IC50 = 15 nM T77537 C6YE8Z 155552072 IC50 = 2133 nM T77537 CXB6U7 155552682 IC50 = 14 nM T77537 C0HUL3 155552710 IC50 = 7.8 nM T77537 CZ9OW5 155558028 IC50 = 14 nM T77537 CPAV79 155559005 IC50 = 55 nM T77537 C4L6HQ 155559509 IC50 = 375 nM T77537 C51IBQ 155560019 IC50 = 7.1 nM T77537 C61NVM 155560973 IC50 = 75 nM T77537 CAC85T 155564156 IC50 = 74 nM T77537 CDAY91 155568779 IC50 = 12 nM T77537 CC29WQ 155568870 IC50 > 10000 nM T77537 CGU74Q 155569301 IC50 = 2.2 nM T77537 D00ERW 44444843 Ki > 1525 nM T77537 D00HVA 11624601 Ki > 3800 nM T77537 D01RHR 71519693 IC50 > 30000 nM T77537 D01VFR 4708 IC50 > 30000 nM T77537 D04PEI 11467730 Ki = 16 nM T77537 D05RPN 11527400 IC50 = 96 nM T77537 D06BJG 71556703 IC50 > 30000 nM T77537 D06WGX 9549184 IC50 > 25000 nM T77537 D0D6MH 11617559 IC50 > 16000 nM T77537 D0E7VO 59627005 IC50 = 72.2 nM T77537 D0GN5Z 5281295 IC50 = 2020 nM T77537 D0J3LR 11634725 Ki > 4000 nM T77537 D0OZ2S 11785878 IC50 > 20000 nM T77537 D0Q0YV 24944925 IC50 = 5495.41 nM T77537 D0Q3NG 11715520 Ki > 3800 nM T77537 D0S7IE 11658882 Ki > 3800 nM T31989 D0L0YG 5280335 IC50 = 1560 nM T31989 D0X6BX 15604015 Ki = 9800 nM T31989 D0DG7E 72735621 IC50 = 5000 nM T31989 D08SUQ 9925886 IC50 = 766000 nM T31989 C3NIO0 282594 IC50 > 100000 nM T31989 C9GF7W 420266 Ki = 6900 nM T31989 CS3X7Z 2936770 IC50 = 62600 nM T31989 C5CF7V 4132571 IC50 = 31300 nM T31989 CLQ2H6 9564003 IC50 = 17100 nM T31989 C8M9ZK 9630678 IC50 = 28510 nM T31989 CSN36K 9660619 IC50 > 100000 nM T31989 CVR8W5 15983462 Ki = 4200 nM T31989 CL7AW8 15983581 Ki = 4200 nM T31989 C9DY1H 45267000 IC50 = 13300 nM T31989 CXP98A 45267876 IC50 = 4380 nM T31989 CJTQ86 45269612 IC50 = 16600 nM T31989 CAZR51 45270448 IC50 = 5730 nM T31989 CU13FG 45271276 IC50 = 7230 nM T31989 C7I1VS 45273014 IC50 = 29200 nM T31989 C7DRY8 46197552 Ki = 500 nM T31989 CE4ZN3 46832080 IC50 = 300 nM T31989 C5T4KE 50916705 Ki = 1500 nM T31989 C5SOT7 53248014 Ki = 4200 nM T31989 C5DMR6 53494962 IC50 = 600 nM T31989 CV8X1J 56840034 Ki = 21000 nM T31989 CK5A3Q 56929818 IC50 = 20 nM T31989 C96HPN 57402828 Ki = 16000 nM T31989 C4R8BS 60149004 Ki = 6000 nM T31989 CUC7B3 66557964 IC50 > 50000 nM T31989 CPR8M7 71449578 Ki = 11000 nM T31989 CH5YO1 71451384 Ki = 43000 nM T31989 C4V8NY 71453197 Ki = 43000 nM T31989 CEC75Q 71458557 Ki = 7000 nM T31989 CH19YZ 71460405 Ki = 8000 nM T31989 CZEM14 71462095 Ki = 29000 nM T31989 C91MOC 71521167 Ki = 8100 nM T31989 CQ7R2F 71627420 IC50 = 1600 nM T31989 CA6MN7 71661218 Ki = 1300 nM T31989 C58SXV 71714682 Ki = 4300 nM T31989 C41HDP 71727564 Ki > 10000 nM T31989 C2JVX0 71727565 Ki = 5200 nM T31989 C6DSB9 71727676 Ki = 1200 nM T31989 CHB2G5 71727800 Ki > 10000 nM T31989 C7HM8J 71812415 IC50 = 40 nM T31989 CQOM26 71812416 IC50 = 40 nM T31989 CIHY54 71812417 IC50 = 20 nM T31989 C1XR2P 71812418 IC50 = 50 nM T31989 CD51FM 71813340 IC50 = 2500 nM T31989 C23DVM 71813341 IC50 = 2500 nM T31989 C4BJU1 71813342 IC50 = 2700 nM T31989 CH75OI 71813505 IC50 = 5700 nM T31989 C0Q7AR 71813506 IC50 = 2900 nM T31989 CO4E5N 71813507 IC50 > 10000 nM T31989 CD5B1M 71813508 IC50 = 3300 nM T31989 CC4MZ3 71813509 IC50 = 3300 nM T31989 CD8G2B 71813510 IC50 > 10000 nM T31989 CNF79K 71813670 IC50 = 1700 nM T31989 C42RXL 71813671 IC50 > 10000 nM T31989 C2YP9U 71813673 IC50 = 1600 nM T31989 CC0Z9Y 71813674 IC50 = 7200 nM T31989 CR20UF 71813675 IC50 = 760 nM T31989 CZ4N6I 71813828 IC50 = 1700 nM T31989 CDG82F 71813829 IC50 = 2200 nM T31989 CA29MU 71813830 IC50 = 3800 nM T31989 CHB8F6 71813831 IC50 > 10000 nM T31989 C8GX0A 71813832 IC50 = 90 nM T31989 CS3U7T 71813975 IC50 = 270 nM T31989 C3WXA8 71813976 IC50 = 250 nM T31989 C6JX4K 71813977 IC50 = 90 nM T31989 C2VB7R 71814309 IC50 = 3700 nM T31989 CNU3R2 71814310 IC50 = 2100 nM T31989 CGI8O9 71814493 IC50 = 1900 nM T31989 CGCK24 71814494 IC50 = 5500 nM T31989 CQ3JF6 71814495 IC50 = 5400 nM T31989 CZNC03 71814496 IC50 = 1700 nM T31989 C8V1TU 71814497 IC50 = 1200 nM T31989 CZVX43 71814498 IC50 = 370 nM T31989 C1ZNP6 71814675 IC50 = 1300 nM T31989 C3Y6GW 71814676 IC50 = 220 nM T31989 CND38P 71814677 IC50 = 430 nM T31989 C4HE3B 71814678 IC50 > 5000 nM T31989 C3HR1T 71814679 IC50 = 150 nM T31989 C6P8KM 71814846 IC50 = 700 nM T31989 C9BJZ6 71814847 IC50 = 3000 nM T31989 CQ62UK 71814848 IC50 = 170 nM T31989 C9FK2A 71814849 IC50 = 4600 nM T31989 CEP2B5 71814850 IC50 = 90 nM T31989 CW1X0Y 71814851 IC50 = 110 nM T31989 CRM17W 71815023 IC50 = 940 nM T31989 C6KC3P 71815024 IC50 > 5000 nM T31989 C8RPW2 71815025 IC50 > 10000 nM T31989 CA68ON 71815026 IC50 = 200 nM T31989 CR8Z6C 71815027 IC50 = 390 nM T31989 CHY3O8 71815028 IC50 > 5000 nM T31989 CBXD42 72735619 IC50 = 5200 nM T31989 CB24ZV 73265274 IC50 = 42600 nM T31989 C3A4KF 73349099 IC50 = 3000 nM T31989 CE7UR8 73353633 Ki > 100000 nM T31989 CF83GY 76325790 IC50 = 21800 nM T31989 C5FDA8 76329372 IC50 = 300000 nM T31989 CIW6T4 89740017 Ki = 10200 nM T31989 C9FM2Y 89740586 Ki = 1200 nM T31989 CFH3S4 89740671 Ki = 14100 nM T31989 CC6MX1 89741221 Ki = 3400 nM T31989 C8ON1V 89741310 Ki = 43000 nM T31989 CCWB78 89741619 Ki = 1100 nM T31989 CBR42S 101913779 IC50 = 6500 nM T31989 C93YFS 118255060 Ki = 6000 nM T31989 CE24JK 118255132 Ki = 1300 nM T31989 C48KEV 118611394 IC50 = 1900 nM T31989 CLQ9R7 118611411 IC50 = 5500 nM T31989 C4F7XM 118734328 Ki = 16500 nM T31989 CN9P8D 118734390 Ki = 1300 nM T31989 CCTD29 122365196 IC50 = 2200 nM T31989 CK16NT 122365197 IC50 = 240 nM T31989 CFD9T6 122365198 IC50 > 30000 nM T31989 C5PH3C 127027128 IC50 = 148 nM T31989 C0EQ9W 127043058 Ki = 11700 nM T31989 CBI8C4 127045038 Ki = 10900 nM T31989 C7JF3L 127045539 Ki = 11000 nM T31989 C54NZV 127045540 Ki = 10300 nM T31989 C5V8PK 127045541 Ki = 9900 nM T31989 C6UA2H 127048340 Ki = 9800 nM T31989 C1EJN8 127048670 IC50 = 81170 nM T31989 CR5J7D 127048671 IC50 = 78690 nM T31989 CI6VY1 127048672 IC50 = 65380 nM T31989 C3T2NZ 127048673 IC50 = 16320 nM T31989 CIOB05 127049002 IC50 > 100000 nM T31989 C51ZEV 127049003 IC50 = 22150 nM T31989 CCH2S3 127049291 IC50 = 44500 nM T31989 C72VGW 127049294 IC50 = 35110 nM T31989 CV1M5H 127049332 IC50 = 43280 nM T31989 CP5TM3 127049333 IC50 = 30230 nM T31989 C32ETI 127049334 IC50 = 26620 nM T31989 C9VJX7 127049335 IC50 = 2170 nM T31989 C0PNK3 127049336 IC50 > 100000 nM T31989 C2MHI6 127049994 IC50 > 100000 nM T31989 CJ51CK 127050232 Ki = 1020 nM T31989 CNV12K 127050290 IC50 > 100000 nM T31989 CJT87U 127050865 IC50 > 100000 nM T31989 CY6MD3 127050920 IC50 = 15080 nM T31989 CI9E4G 127050921 IC50 = 23830 nM T31989 CRCG86 127050922 IC50 = 15640 nM T31989 CO0M4W 127050923 IC50 = 44540 nM T31989 CVIN74 127050924 IC50 = 22590 nM T31989 CMB5C6 127051152 Ki = 900 nM T31989 C0NXA4 127051153 Ki = 980 nM T31989 CTSP67 127051186 IC50 = 17790 nM T31989 CJ3KN5 127051492 IC50 > 100000 nM T31989 CD4P9L 127051493 IC50 > 100000 nM T31989 C8JW6R 127051494 IC50 = 13840 nM T31989 CD5FY0 127051495 IC50 > 100000 nM T31989 C5C2UN 127051496 IC50 > 100000 nM T31989 CP9O2Q 127051497 IC50 = 11400 nM T31989 C4U3VW 127051810 IC50 = 68550 nM T31989 CDV4I7 127052117 IC50 > 100000 nM T31989 C5W3BG 127052118 IC50 = 40580 nM T31989 C3W2BY 127052119 IC50 = 19530 nM T31989 C6B5ML 127052120 IC50 = 8700 nM T31989 CKB92N 127052121 IC50 > 100000 nM T31989 CFZ6M0 127052140 Ki = 980 nM T31989 CFQ63S 127052141 Ki = 3800 nM T31989 C1XRW2 127052719 IC50 = 98900 nM T31989 CZY17D 127052720 IC50 > 100000 nM T31989 CB6JF5 127052721 IC50 > 100000 nM T31989 CV0LF4 127052728 IC50 > 100000 nM T31989 C63CWH 127052729 IC50 = 4600 nM T31989 C7BMU9 127052730 IC50 > 100000 nM T31989 CL02DX 127052731 IC50 > 100000 nM T31989 CH8PE9 127052732 IC50 > 100000 nM T31989 CG4KH8 127052733 IC50 = 10150 nM T31989 CZWF94 127052734 IC50 > 100000 nM T31989 C58VJN 127053007 IC50 = 58790 nM T31989 CCJ71P 127053008 IC50 = 67370 nM T31989 C0U1SE 127053009 IC50 = 61200 nM T31989 CW3EN2 127053010 IC50 = 62170 nM T31989 C9A7BH 134812833 Ki = 370 nM T31989 C54FXD 134957362 IC50 > 10000 nM T31989 C0YDR9 137553159 IC50 = 145 nM T31989 CJHA89 137631941 IC50 > 100000 nM T31989 CG46PI 137632626 IC50 < 1.7 nM T31989 CYB4Z5 137633994 IC50 = 840 nM T31989 CF8T9O 137634221 IC50 = 164 nM T31989 CAW7X5 137634618 IC50 = 7230 nM T31989 CV65UW 137634788 IC50 = 465 nM T31989 CM9X6B 137635845 IC50 = 21000 nM T31989 CU65BI 137636078 IC50 > 100000 nM T31989 CX8DI3 137636195 IC50 = 2100 nM T31989 CC30PZ 137638678 Ki = 170 nM T31989 C2ZEL8 137639097 IC50 = 8300 nM T31989 CB3D4T 137641685 IC50 > 30000 nM T31989 C9FID2 137642040 IC50 > 30000 nM T31989 C1T8DM 137642521 IC50 > 100000 nM T31989 CSQH31 137643140 IC50 < 1.7 nM T31989 C9W3NK 137643775 IC50 = 164 nM T31989 CDH76B 137644043 IC50 = 1700 nM T31989 COMC94 137646013 Ki = 170 nM T31989 CAME30 137646035 IC50 = 46000 nM T31989 C51LSX 137647661 IC50 = 670 nM T31989 CQLJ28 137649154 IC50 > 30000 nM T31989 C3KN9J 137649735 IC50 = 780 nM T31989 CDT06A 137649743 Ki = 90 nM T31989 CP63XR 137650218 Ki = 390 nM T31989 CQ2M6U 137650955 IC50 = 443 nM T31989 C7QT3K 137651095 Ki = 900 nM T31989 C9KMW8 137651971 IC50 = 1900 nM T31989 CF0Q3L 137652248 Ki = 90 nM T31989 CA84YU 137653104 IC50 = 1300 nM T31989 CABF71 137653763 Ki = 250 nM T31989 CLF8M0 137657883 IC50 = 2.4 nM T31989 CKH03X 137657977 IC50 = 35100 nM T31989 CX63PI 137658079 IC50 = 3900 nM T31989 CHUZ37 137658235 IC50 > 30000 nM T31989 C8P7TG 137659208 IC50 = 9400 nM T31989 CH2AN7 137660780 IC50 = 39600 nM T31989 CKOQ53 137660812 IC50 = 460 nM T31989 CK7LE0 137661361 IC50 = 560 nM T31989 CK3D2P 154699447 IC50 = 16 nM T31989 C0QY4W 154699448 IC50 = 41 nM T31989 C8NI1W 154699449 IC50 = 17 nM T31989 CYUT01 154699450 IC50 = 31 nM T31989 C1CAT9 155517174 IC50 = 902 nM T31989 CNB93E 155519701 IC50 = 119 nM T31989 CSGJ75 155523497 IC50 = 151 nM T31989 C89YXV 155524292 EC50 = 59 nM T31989 CF78NS 155524444 EC50 = 50 nM T31989 CTP85C 155525319 IC50 = 49 nM T31989 CZ82OI 155525383 IC50 = 412 nM T31989 CXB1Q7 155528975 EC50 = 37 nM T31989 CON56I 155531486 EC50 = 146 nM T31989 C0MC9O 155535418 IC50 = 35 nM T31989 C31DCI 155536233 EC50 = 84 nM T31989 CC62JR 155536715 IC50 = 143 nM T31989 C0ITD5 155555664 IC50 = 55 nM T31989 CR96ED 155557208 IC50 = 1120 nM T31989 CZ06PJ 155564368 EC50 = 73 nM T31989 CQL4F1 155564588 IC50 = 26 nM T31989 CC9F8Z 155569662 EC50 = 32 nM T31989 D00YNY 753704 Ki = 6700 nM T31989 D05SLY 44815217 IC50 = 10000 nM T31989 D08SND 66577038 Ki = 3.6 nM T31989 D0H2LN 71458556 Ki = 16500 nM T31989 D0M9DT 5282309 Ki = 12000 nM T31989 D0P5TI 58441401 IC50 > 1000 nM T31989 D0TC4I 45483175 Ki = 31000 nM T91558 C81ITX 85473309 IC50 = 46 nM T91558 C4O1LQ 85473438 IC50 = 0.012 nM T91558 C81ILP 138471783 IC50 = 290 nM T91558 CEK6B1 139300630 IC50 > 10000 nM T76904 D0J1VY 5281081 IC50 = 386 nM T76904 D0Y7PG 4659569 IC50 < 1 nM T76904 D01SGK 135565903 Ki = 1 nM T76904 D0E4WF 439176 Ki > 5400000 nM T76904 C1KG9Z 6792 IC50 = 6309.57 nM T76904 C7GLB3 2805447 Ki = 7900 nM T76904 CC4O6E 5152843 Ki = 251000 nM T76904 CLRD65 7147386 Ki = 6300 nM T76904 C0OE3C 10397916 IC50 = 18000 nM T76904 CF35YR 12468238 IC50 = 3400 nM T76904 C8C5OA 13130143 IC50 = 1700 nM T76904 CJLU70 14602319 IC50 > 10000 nM T76904 CK3C5U 15982971 Ki < 1 nM T76904 C3LM8W 19616700 Ki = 25000 nM T76904 C0I6QS 45266258 Ki = 5800000 nM T76904 C7Z3EI 45266259 Ki = 800000 nM T76904 CJO7Y5 45266260 Ki = 800000 nM T76904 CX5KA8 45266261 Ki = 6000000 nM T76904 C6OWN4 45266294 Ki = 500000 nM T76904 CSQW23 45588801 IC50 > 10000 nM T76904 C0OH4L 46865888 Ki = 17 nM T76904 C4JUD1 46865889 Ki = 1.6 nM T76904 CU9N6Q 46884860 Ki = 2.2 nM T76904 CE26QR 46884861 Ki = 9.2 nM T76904 CWF6J3 46884905 Ki = 1.3 nM T76904 CD8WZ0 46884906 Ki = 1.1 nM T76904 CE25JB 46884907 Ki = 10.2 nM T76904 CHI9F2 46884908 Ki = 17 nM T76904 CBZ6E7 46884909 Ki = 10.6 nM T76904 C6J5ZS 46884939 Ki = 16.6 nM T76904 C3FN6H 46884940 Ki = 6 nM T76904 CA03ZI 53379376 IC50 = 200 nM T76904 CVKW93 53379379 IC50 = 61 nM T76904 CNS4P0 53380912 IC50 = 47 nM T76904 CY7P2A 67405675 IC50 = 128 nM T76904 CJIM75 67418555 IC50 = 53 nM T76904 CGK4V8 67419355 IC50 = 87 nM T76904 CF80AB 67419505 IC50 = 3020 nM T76904 CBO31T 69929269 IC50 = 170 nM T76904 CHLG32 69931826 IC50 = 35 nM T76904 C5FVM1 69932256 IC50 = 706 nM T76904 CEDU65 69932313 IC50 = 680 nM T76904 C0W4YT 69932481 IC50 = 101 nM T76904 C9I8JN 69932517 IC50 = 1500 nM T76904 CXO59G 69932543 IC50 > 5000 nM T76904 C6C3SV 69932581 IC50 = 2400 nM T76904 C0WFN4 71395955 IC50 = 19.95 nM T76904 CMA72V 89466901 IC50 = 84 nM T76904 CQG3M5 89467005 IC50 = 55 nM T76904 CO1F2M 118736597 IC50 = 400 nM T76904 CVD30G 118736600 IC50 > 10000 nM T76904 CFCS69 118736601 IC50 = 4500 nM T76904 C8CNJ1 118736602 IC50 = 5800 nM T76904 C5SB8X 118736603 IC50 = 5500 nM T76904 C0FIS1 118736604 IC50 = 160 nM T76904 CJCQ91 118736605 IC50 = 140 nM T76904 CZ1FH9 118736606 IC50 = 140 nM T76904 CM2T4P 118736607 IC50 = 88 nM T76904 CBLT83 118736608 IC50 = 57 nM T76904 CDZ9V5 118736609 IC50 = 1900 nM T76904 CZ85HC 118736610 IC50 = 13000 nM T76904 CF0Z7Q 122439995 IC50 = 1.995 nM T76904 C1PE9K 122440001 IC50 = 3.981 nM T76904 CQ9FG1 122440007 IC50 = 199.53 nM T76904 CRV7L1 122440022 IC50 = 10 nM T76904 C9TP2N 122440029 IC50 = 19.95 nM T76904 CKS61V 122440030 IC50 = 79.43 nM T76904 CB54TV 122440031 IC50 = 7.943 nM T76904 C5R2JV 122441915 IC50 = 6.31 nM T76904 C4OJ6D 122441945 IC50 = 316.23 nM T76904 C6NL1P 122441948 IC50 > 10000 nM T76904 C7A5TQ 122441954 IC50 = 1584.89 nM T76904 CI65KH 122441965 IC50 = 6.31 nM T76904 CPLQ64 122441976 IC50 = 63.1 nM T76904 C85YVR 122441981 IC50 = 1258.93 nM T76904 C92VAF 122442004 IC50 = 19.95 nM T76904 C36XNY 122442007 IC50 = 3.162 nM T76904 C4WVK0 122442029 IC50 = 3.981 nM T76904 CD9IE5 122442045 IC50 > 10000 nM T76904 CA35KX 122442051 IC50 = 1.995 nM T76904 C7KTJ8 127046300 IC50 = 456 nM T76904 CJ6WA2 127046783 IC50 > 5000 nM T76904 C0ZWY6 127047871 IC50 = 962 nM T76904 CB5I2N 127047926 IC50 = 1667 nM T76904 CQU46R 127048055 IC50 = 826 nM T76904 C8F2XG 127048056 IC50 = 672 nM T76904 C7VJ3D 127048057 IC50 = 574 nM T76904 C8DT5E 127048058 IC50 = 49.5 nM T76904 C0OY3S 127050334 IC50 = 179 nM T76904 CTH9J4 127050335 IC50 = 54 nM T76904 CQA4M8 127050621 IC50 = 648 nM T76904 CK0DI2 129165296 IC50 = 50 nM T76904 C83LIY 129165316 IC50 = 10 nM T76904 C8BOL3 129165356 IC50 = 10 nM T76904 CFGM98 129165376 IC50 = 220 nM T76904 C3H8LN 129165377 IC50 = 60 nM T76904 CF67NH 129165444 IC50 = 630 nM T76904 CG3OP9 129165448 IC50 = 63 nM T76904 CJGE94 129165458 IC50 = 40 nM T76904 CDT58P 129165460 IC50 = 16 nM T76904 C0F7CK 129165469 IC50 = 400 nM T76904 CHZ7N2 129165491 IC50 = 250 nM T76904 CXU3W9 129165493 IC50 = 6.3 nM T76904 CJ51DV 129165494 IC50 = 38 nM T76904 CY5X3U 129165527 IC50 = 100 nM T76904 CI0C1P 129165534 IC50 = 13 nM T76904 C1DPO0 129165543 IC50 = 40 nM T76904 CTUA67 129165554 IC50 = 50 nM T76904 CO0VS6 129165556 IC50 = 40 nM T76904 CW2S3J 129165564 IC50 = 450 nM T76904 C8OC4X 136934927 IC50 = 2100 nM T76904 CK0ZP6 140931610 IC50 = 6300 nM T76904 C48UMS 145949230 IC50 = 1584.89 nM T76904 CD3M0U 145950392 IC50 > 10000 nM T76904 CVR04X 145951510 IC50 = 251.19 nM T76904 C7SMJ2 145956792 IC50 = 3981.07 nM T76904 CHO0E4 155518634 IC50 = 1600 nM T76904 C6ATD2 155523978 IC50 = 2000 nM T76904 C3B0SN 155543374 IC50 > 10000 nM T76904 CCNW79 155543901 IC50 = 2000 nM T76904 CQLM48 155562927 IC50 > 10000 nM T76904 D0FO2B 1923 IC50 = 3162.28 nM T31424 D01AZG 5073 Ki = 1.8 nM T31424 D01JUF 5775 Ki = 5 nM T31424 D03SKR 2803 Ki = 3.8 nM T31424 D04PHC 5816 Ki = 5 nM T31424 D05DVP 5717 IC50 > 10000 nM T31424 D06OFS 68712 Ki = 180 nM T31424 D07MOX 439260 Ki = 30 nM T31424 D09EBS 4636 Ki = 2.2 nM T31424 D0D1AL 3559 Ki > 5000 nM T31424 D0E9PK 4810 Ki = 75 nM T31424 D0H4JM 8969 Ki = 0.4 nM T31424 D0H7KF 5002 Ki = 87 nM T31424 D0MT0M 2216 EC50 = 1.9 nM T31424 D0O6IU 6041 Ki = 390 nM T31424 D0O6IZ 4436 IC50 = 0.0011 nM T31424 D0R1JV 60854 Ki = 390 nM T31424 D0T0KA 4474 IC50 > 10000 nM T31424 D0T6QX 5736 Ki = 180 nM T31424 D0V4QS 135398745 Ki = 140 nM T31424 D0WV3U 4893 Ki = 34 nM T31424 D0X6BV 6918314 IC50 = 6000 nM T31424 D0Y4DY 5709 Ki > 500 nM T31424 D0Z1RV 135398737 Ki = 51 nM T31424 D0F2ML 68602 EC50 = 3 nM T31424 D02FNU 56971 IC50 = 1000 nM T31424 D06DZI 107780 Ki < 1000 nM T31424 D0BC6Q 9837551 Ki = 1.2 nM T31424 D0OS6O 60149 Ki = 1680 nM T31424 D0ZG9N 132337 Ki > 10000 nM T31424 CZUI83 2769 IC50 = 4500 nM T31424 C32BCH 4656 IC50 = 1.5 nM T31424 CY1OB3 24484 Ki = 416.87 nM T31424 CU86VK 54459 Ki = 51.29 nM T31424 COTZ60 68601 IC50 = 3300 nM T31424 C4X7HB 72016 Ki = 51.29 nM T31424 CB17UR 127901 Ki = 1200 nM T31424 CUDB20 127904 Ki = 1000 nM T31424 C2H1VA 131829 Ki = 6 nM T31424 C3LG9C 132110 IC50 = 0.0034 nM T31424 CZL87W 133999 IC50 > 10000 nM T31424 C9NW0U 135152 Ki = 48 nM T31424 CCP43U 146762 EC50 = 1200 nM T31424 CKFG02 172745 Ki = 700 nM T31424 CA9XQ1 183823 Ki = 230 nM T31424 CF4V5Q 185076 EC50 = 0.26 nM T31424 C9JR4O 271890 Ki = 269.15 nM T31424 CUN08L 280604 Ki = 363.08 nM T31424 CX9V6O 411679 EC50 = 30400 nM T31424 C91HBL 541604 Ki = 9 nM T31424 C54QJC 3086247 Ki = 3.1 nM T31424 CN3F2W 3086489 EC50 = 141000 nM T31424 CZHG83 3416533 Ki = 2215 nM T31424 CC9V5K 4013695 Ki >= 1000 nM T31424 C6AML5 5288606 Ki = 220 nM T31424 CPR2E4 9549064 Ki = 205 nM T31424 CCSN93 9800737 IC50 = 7000 nM T31424 C8XGV3 9804849 IC50 = 1.3 nM T31424 CGJB47 9816035 Ki > 500 nM T31424 CH7U3C 9816604 Ki = 1320 nM T31424 CD6NB7 9816895 Ki > 10000 nM T31424 C95BXW 9823464 IC50 = 900 nM T31424 CRW5N0 9837525 Ki > 500 nM T31424 CJ8LT7 9848518 IC50 > 10000 nM T31424 C3YSQ5 9859238 Ki = 46 nM T31424 C7EZ2L 9859861 Ki > 7800 nM T31424 CT2C6K 9870702 IC50 > 10000 nM T31424 CPI8G9 9881158 Ki = 5.2 nM T31424 C6CZ3G 9906777 IC50 > 10000 nM T31424 CO7BK6 9909648 Ki = 181 nM T31424 CR9KM0 9921064 Ki = 300 nM T31424 CH5D3J 9928343 IC50 > 10000 nM T31424 CQIU94 9978693 IC50 = 2000 nM T31424 CDG59F 9997892 Ki = 1584.89 nM T31424 CWMF43 10019859 Ki = 57.54 nM T31424 C5MZ6I 10042547 Ki > 2500 nM T31424 CQ9O8W 10105615 EC50 = 32992 nM T31424 CNA8W3 10130620 Ki = 1120 nM T31424 CL53TD 10176639 Ki > 10000 nM T31424 C6S2RA 10198552 Ki = 0.25 nM T31424 C9FDM0 10263774 Ki = 1400000 nM T31424 C3NGO6 10332138 Ki = 1400000 nM T31424 C5BME0 10374995 Ki > 10000 nM T31424 CS2DN8 10376336 EC50 = 375 nM T31424 C8OZ2X 10401405 Ki > 1000000 nM T31424 CW9HZ1 10401566 Ki = 1000 nM T31424 C7LGR3 10420352 Ki = 66 nM T31424 C7FDR9 10474619 Ki > 2240 nM T31424 CWC3X7 10658207 IC50 = 97700 nM T31424 CND1W5 11390143 EC50 = 45300 nM T31424 C16TWK 11508052 IC50 > 10000 nM T31424 CXWO08 11522273 IC50 > 10000 nM T31424 CQ08DH 11539632 IC50 = 0.25 nM T31424 CTCW08 11680583 Ki > 1000000 nM T31424 CN9H3J 11820372 EC50 = 18 nM T31424 CB9YK4 12406841 IC50 = 10000 nM T31424 CIUR20 12699315 Ki > 1949 nM T31424 C8SG1D 13041565 Ki = 645.65 nM T31424 C3NC7P 13338337 Ki = 232 nM T31424 CRN3S9 13387299 Ki = 77 nM T31424 CPA2O9 13387301 Ki = 10.7 nM T31424 CIDB37 13387304 Ki = 670 nM T31424 CXS0R8 13387308 Ki = 13000 nM T31424 CWVT29 13392482 Ki = 6.1 nM T31424 C1LXY9 13473217 Ki = 25 nM T31424 C9BQ5D 13473220 Ki = 7 nM T31424 CLYK03 13538579 Ki = 15 nM T31424 CES6X1 13538583 Ki = 470 nM T31424 C36HGR 13538585 Ki = 520 nM T31424 CV6FD5 13720763 Ki = 18 nM T31424 CIH1X9 13805911 IC50 = 2000 nM T31424 C8N6SI 14442245 IC50 >> 1000 nM T31424 CG59NT 14548271 IC50 > 1000 nM T31424 CX65HY 14548274 IC50 = 10000 nM T31424 C40LIM 14548276 IC50 >> 1000 nM T31424 C3AB0I 14548281 IC50 > 1000 nM T31424 CF4UR7 14548283 IC50 >> 1000 nM T31424 C60PQZ 14548284 IC50 > 1000 nM T31424 C4T3VO 14548286 IC50 >> 10000 nM T31424 CKI6C0 14548290 IC50 > 100000 nM T31424 CS9Q1A 14920657 Ki = 616.6 nM T31424 C7JV1Z 15054187 Ki > 100000 nM T31424 C5RM1O 15054189 Ki = 55 nM T31424 C7Z4YC 15054190 Ki > 100000 nM T31424 CKVQ30 15054191 Ki > 100000 nM T31424 CEBL08 15054192 Ki > 100000 nM T31424 C6US3O 15711850 Ki = 358 nM T31424 C5PO3N 15711869 Ki = 360 nM T31424 CW9O3C 17755236 EC50 = 355000 nM T31424 CC39VZ 17755537 Ki = 100 nM T31424 CLK2Q9 17755543 EC50 = 2760 nM T31424 C02MUZ 17755548 Ki = 18.2 nM T31424 CSK7W1 19032629 Ki = 5248.07 nM T31424 C6V4GU 20447226 Ki = 338 nM T31424 C7FZ8G 21539587 Ki = 400000 nM T31424 CMZL78 21584293 Ki = 28000 nM T31424 C0BL3K 23499169 Ki = 95.5 nM T31424 CNU2X4 23725134 IC50 > 1000 nM T31424 C72CMN 24749577 Ki = 3928 nM T31424 C0I2HU 24769156 Ki = 150 nM T31424 C3JSR4 24794436 IC50 > 1000 nM T31424 C4OTN7 25209507 Ki = 53.7 nM T31424 CJ5P2S 25209509 Ki = 177.83 nM T31424 CV36LQ 25209671 Ki = 112.2 nM T31424 CUQB19 25209673 Ki = 75.86 nM T31424 CX94FK 25209826 Ki = 41.69 nM T31424 CQ59WF 25209828 Ki = 263.03 nM T31424 C35PDJ 29181446 EC50 = 42200 nM T31424 C9RY0G 29922170 Ki = 10000 nM T31424 C1FRU8 44288600 IC50 = 6400 nM T31424 C7AJ3B 44293793 Ki = 5300 nM T31424 CYUA79 44293794 Ki = 180 nM T31424 CJ7F1Y 44313718 Ki = 6309.57 nM T31424 C7RO6Z 44313966 Ki = 1.585 nM T31424 CBO94A 44340588 Ki = 3900000 nM T31424 CAN1E0 44340624 Ki = 2900000 nM T31424 C2UC0K 44375762 Ki = 1380.38 nM T31424 CHYN70 44377985 IC50 = 0.61 nM T31424 C2P7TG 44405404 Ki > 1000000 nM T31424 C4YUS1 44405471 Ki > 1000000 nM T31424 C0QHU8 44405493 Ki > 1000000 nM T31424 CFH35N 44405494 Ki > 1000000 nM T31424 C9V1NR 44405495 Ki = 1100 nM T31424 C4AXG5 44405498 Ki = 1200 nM T31424 CA3IP7 44405499 Ki = 3900 nM T31424 CQJ26O 44405513 Ki = 36000 nM T31424 C0EXA1 44407083 IC50 > 10000 nM T31424 CG3OY5 44427965 Ki = 1659.59 nM T31424 C8UON6 44474625 IC50 > 10000 nM T31424 C6HVU1 44474629 IC50 > 10000 nM T31424 CE2Z8S 44474631 IC50 > 1000 nM T31424 C8LA4W 44474797 IC50 > 1000 nM T31424 C52OLJ 44570725 EC50 = 38700 nM T31424 C38XRH 45262914 IC50 = 0.016 nM T31424 C9R2ZY 45262937 IC50 = 0.034 nM T31424 C6PJD1 45263619 Ki = 467.74 nM T31424 C8WF5L 45265388 IC50 = 0.014 nM T31424 C0U8HZ 45265408 IC50 = 0.12 nM T31424 CX1WO9 45265432 IC50 = 0.26 nM T31424 C8A9ZJ 45265927 Ki = 1071.52 nM T31424 CD5H2X 45483622 IC50 > 10000 nM T31424 C8BK9U 52944141 EC50 = 16000 nM T31424 CQ18HL 56837266 Ki = 1949.84 nM T31424 CC9D5Z 56837268 Ki = 181.97 nM T31424 CW41AD 56840511 Ki = 1995.26 nM T31424 C1FGI9 56840512 Ki = 2398.83 nM T31424 CJZ14R 56840513 Ki = 933.25 nM T31424 C7RN9D 56840514 Ki = 165.96 nM T31424 C9WZ5L 66570978 Ki > 10000 nM T31424 C6PL9B 66571028 Ki > 10000 nM T31424 CAQ2T8 66571029 Ki > 10000 nM T31424 CT3NO0 66571030 Ki > 10000 nM T31424 C7QT9R 66571031 Ki > 10000 nM T31424 C9U7YI 66571032 Ki > 10000 nM T31424 CNID83 66571033 Ki > 10000 nM T31424 CFE96S 70031156 Ki = 10000 nM T31424 C3DY6Q 70980100 Ki > 10000 nM T31424 CA34VD 70980467 Ki > 10000 nM T31424 CDI84E 71450922 IC50 > 10000 nM T31424 C73EGZ 89964574 Ki = 10000 nM T31424 CW50FJ 101836086 Ki = 39810.72 nM T31424 CZ2O9K 118730388 Ki = 75857.76 nM T31424 CILU63 118730390 Ki = 162181.01 nM T31424 C2PTS4 118730391 Ki = 6606.93 nM T31424 C1ZVG5 118730392 Ki = 10715.19 nM T31424 C5FO1D 118730393 Ki = 2691.53 nM T31424 CB9Q7A 118730395 Ki = 446.68 nM T31424 CK24SH 118730399 Ki = 562.34 nM T31424 CJR8T1 118730401 Ki = 389.05 nM T31424 CARN54 118730403 Ki = 537.03 nM T31424 C19WRG 118730405 Ki = 2238.72 nM T31424 C6DTU2 118730499 Ki = 74.13 nM T31424 CU45ZK 118730502 Ki = 954.99 nM T31424 C6SF7J 118730504 Ki = 177.83 nM T31424 CC5P4U 118730506 Ki = 4168.69 nM T31424 CC6NA7 118730508 Ki = 6165.95 nM T31424 CLH27O 118730510 Ki = 1479.11 nM T31424 C8EG4M 118730512 Ki = 478.63 nM T31424 CNEJ15 118730513 Ki = 524.81 nM T31424 CZET94 118730516 Ki = 213.8 nM T31424 C5KFB7 118730519 Ki = 549.54 nM T31424 CL51OZ 118730521 Ki = 4466.84 nM T31424 C39FAJ 118730523 Ki = 46773.51 nM T31424 CDMU26 118730525 Ki = 32359.37 nM T31424 CI9C3V 118730527 Ki = 31622.78 nM T31424 C9GE4M 118730529 Ki = 5011.87 nM T31424 C3ROW1 127046249 EC50 = 7.9 nM T31424 CA4HX1 127047326 EC50 = 3600 nM T31424 C3RI9A 134134855 Ki = 7079.46 nM T31424 CQX7Z9 134137282 Ki = 1412.54 nM T31424 CMN2V1 134145891 Ki = 724.44 nM T31424 C2GZM7 134147006 Ki = 8912.51 nM T31424 C9P8MT 134147299 Ki = 10232.93 nM T31424 C73JQM 134151527 Ki = 281.84 nM T31424 CQ8C3K 134151763 Ki = 8511.38 nM T31424 C27VRU 134151905 Ki = 1548.82 nM T31424 CB2T0I 134151989 Ki = 10232.93 nM T31424 CW87FZ 134153595 Ki = 4365.16 nM T31424 CW7Q3A 134154917 Ki = 229.09 nM T31424 CSM40A 134155182 Ki = 7762.47 nM T31424 CA3SB0 134155234 Ki = 12022.64 nM T31424 CDQ58J 134156245 Ki = 3162.28 nM T31424 CPB9I7 134156428 Ki = 5128.61 nM T31424 C5OU1T 135409492 Ki > 10000 nM T31424 C4PM9W 135515431 Ki = 783 nM T31424 CSX34L 141469440 Ki = 751 nM T31424 CA4SD5 145960502 Ki > 100000 nM T31424 CK9ME6 145961067 Ki = 1968 nM T31424 CZG31U 145961142 Ki = 706 nM T31424 C5H3JO 145961439 Ki = 1205 nM T31424 C3R8QY 145961538 Ki = 87.9 nM T31424 CK6Y8D 145961752 Ki > 100000 nM T31424 CODR71 145961869 Ki = 9086 nM T31424 CLU0C4 145962173 Ki = 733 nM T31424 CD95LT 145962271 Ki = 2215 nM T31424 CA74EL 145962555 Ki = 66530 nM T31424 CV5Z9D 145962777 Ki = 156 nM T31424 C2BL1O 145962999 Ki > 100000 nM T31424 CI5D9Z 145963040 Ki = 30150 nM T31424 C9D3NQ 145963342 Ki = 31.3 nM T31424 CG0J8H 145963373 Ki = 1198 nM T31424 D00GEE 92766 IC50 = 211000 nM T31424 D01SRS 15407445 Ki = 31000 nM T31424 D02TQC 14928441 Ki = 41 nM T31424 D04AZE 3277600 Ki < 1000 nM T31424 D05KUM 135446209 Ki = 1000 nM T31424 D06UBB 123981 Ki = 16.7 nM T31424 D08KLH 108094 Ki = 0.912 nM T31424 D09CUJ 1862 Ki = 12 nM T31424 D09NXU 10513867 IC50 = 14300 nM T31424 D09PIF 142067 Ki = 7.8 nM T31424 D0C9DC 123920 Ki = 21 nM T31424 D0F3AR 9991628 IC50 = 215400 nM T31424 D0H1WR 5226 Ki = 100000 nM T31424 D0K3UL 9796720 Ki = 400 nM T31424 D0N7UE 10198248 Ki = 41 nM T31424 D0P5PW 132111 EC50 = 9 nM T31424 D0Z7EA 643606 Ki = 0.1 nM T19368 D0T9TJ 3034010 IC50 = 6 nM T19368 D02NHW 2810413 IC50 = 130 nM T19368 CBS6H4 2734352 IC50 = 11000 nM T19368 C03TJI 2809636 IC50 > 50000 nM T19368 CY27ZP 2810411 IC50 = 200 nM T19368 C57UNE 4100861 IC50 = 2000 nM T19368 CP06OA 4197991 IC50 = 320 nM T19368 C69IFT 4589191 IC50 = 470 nM T19368 CEB78U 9795865 IC50 = 1600 nM T19368 C0BA2K 11989651 IC50 = 1000 nM T19368 C6D5JN 18172813 IC50 = 200 nM T19368 CZ7H1I 18525723 IC50 = 1300 nM T19368 C1Q3RG 25181478 IC50 = 130 nM T19368 CRS28P 25181479 IC50 = 130 nM T19368 CU9DL7 25265105 IC50 = 160 nM T19368 C6HJ9P 44569312 IC50 > 50000 nM T19368 CHD61W 44569313 IC50 = 2500 nM T19368 CW9N3U 44569314 IC50 > 50000 nM T19368 C79JKE 44569315 IC50 > 50000 nM T19368 C9GNB0 44569316 IC50 > 50000 nM T19368 CQ9ON6 44569336 IC50 > 50000 nM T19368 CKU51O 44569369 IC50 > 50000 nM T19368 CAZ6K9 44569828 IC50 = 130 nM T19368 CNSZ31 44569829 IC50 > 50000 nM T19368 C7Y8KS 44569830 IC50 = 60 nM T19368 CM15GN 44569863 IC50 > 50000 nM T19368 CZ6TW9 44569864 IC50 > 50000 nM T19368 CV62UJ 44569865 IC50 = 25000 nM T19368 C2Y5AC 44569903 IC50 = 1300 nM T19368 C9TPW6 44569904 IC50 = 250 nM T19368 CF90QM 44569905 IC50 = 1000 nM T19368 CMR30J 44569906 IC50 = 300 nM T19368 C93ZJI 46739726 IC50 = 1700 nM T19368 C1ND3M 54704622 IC50 = 1760 nM T19368 CQ76TF 57391265 IC50 = 2800 nM T19368 C7K6JT 57391611 IC50 = 1000 nM T19368 CA4F1U 57394765 IC50 = 12800 nM T19368 CP03HF 57394766 IC50 = 1100 nM T19368 CTC2Q5 57396517 IC50 = 5000 nM T19368 CR8E0J 57396518 IC50 = 1100 nM T19368 C8P7XU 57396519 IC50 = 1100 nM T19368 C4XS7C 57398310 IC50 = 4500 nM T19368 CTAG79 57399970 IC50 = 5000 nM T19368 CW5DX2 57399971 IC50 = 3100 nM T19368 C1X8DV 57401757 IC50 = 11000 nM T19368 CL3O8E 57401758 IC50 = 300000 nM T19368 C3WCR8 57403489 IC50 = 35000 nM T19368 C3PJ4N 62709758 IC50 = 1010 nM T19368 C54WKD 70800861 IC50 = 400 nM T19368 CLAY09 71515507 IC50 = 5.4 nM T19368 CCZ6O5 71715027 IC50 = 14 nM T19368 CJL85Y 71715030 IC50 = 39 nM T19368 CFQ2A1 71768949 IC50 = 91 nM T19368 CJ0SE5 72735958 IC50 > 10000 nM T19368 C4C2NF 72735959 IC50 = 1960 nM T19368 CRH31E 72735960 IC50 = 184 nM T19368 C9GPA3 72735961 IC50 = 259 nM T19368 C3CT9N 72735962 IC50 = 25 nM T19368 CPED61 72736167 IC50 = 372 nM T19368 C0DCX2 72736168 IC50 = 236 nM T19368 C59NRU 72736169 IC50 = 131 nM T19368 CH1M8V 72736170 IC50 = 236 nM T19368 CS7L8X 72736171 IC50 = 156 nM T19368 CYQ56E 72736172 IC50 = 366 nM T19368 CA5IR2 72736173 IC50 = 110 nM T19368 CA3CX9 72736345 IC50 = 130 nM T19368 C29JMD 72736346 IC50 = 120 nM T19368 C8WK3T 72736347 IC50 = 214 nM T19368 C6E9WO 72736348 IC50 = 88 nM T19368 CSZ58X 72736349 IC50 = 570 nM T19368 C52PVL 72736350 IC50 = 499 nM T19368 CF4HQ3 72736351 IC50 = 551 nM T19368 CYV7G6 72736519 IC50 = 659 nM T19368 CO5BM8 72736520 IC50 = 209 nM T19368 C0DS1N 72736521 IC50 > 10000 nM T19368 C62FEZ 72736522 IC50 > 10000 nM T19368 C27LXW 72736523 IC50 = 1946 nM T19368 C6JI0S 72944619 IC50 < 10 nM T19368 CNVF95 72944930 IC50 < 10 nM T19368 C7KH2Y 73351940 IC50 = 23 nM T19368 C8MX6K 73507100 IC50 < 10 nM T19368 CAVZ58 76317178 IC50 = 33335 nM T19368 CUF96M 76331799 IC50 = 4 nM T19368 C6NM0V 86728184 IC50 = 264 nM T19368 CUPF79 89489281 IC50 = 29 nM T19368 C5XD9L 89489291 IC50 = 88 nM T19368 CDS9O3 89489300 IC50 = 190 nM T19368 C2PTZ5 89489304 IC50 = 59 nM T19368 CKFJ49 89489363 IC50 = 3.6 nM T19368 C58DAC 89489375 IC50 = 2950 nM T19368 CA7DM1 89489436 IC50 = 3520 nM T19368 CI0KQ8 89489635 IC50 < 10 nM T19368 CSWA39 89862351 IC50 = 80 nM T19368 C3L0JQ 89862354 IC50 = 26 nM T19368 CH4GO3 89922162 IC50 < 10 nM T19368 CCJL63 89932422 IC50 < 10 nM T19368 CN7HP3 89961969 IC50 = 5 nM T19368 C9Y3FO 89961977 IC50 = 10 nM T19368 C08TZK 89963108 IC50 = 10 nM T19368 C58USE 89967420 IC50 = 10 nM T19368 C46HRF 90047761 IC50 = 30 nM T19368 CIF9T4 90056613 IC50 = 2700 nM T19368 C53GVA 90056826 IC50 < 10 nM T19368 CCRM78 90056902 IC50 = 10 nM T19368 CTHG91 90057548 IC50 < 10 nM T19368 CK3H2R 90057735 IC50 = 10 nM T19368 C1FS2D 90057739 IC50 = 10 nM T19368 CWO03Y 90057968 IC50 = 100 nM T19368 C76WRO 90078999 IC50 < 10 nM T19368 CC7B2S 90079032 IC50 < 10 nM T19368 CET4R6 90082284 IC50 = 340 nM T19368 C5UP1L 90302077 IC50 = 5830 nM T19368 CWVK69 90302407 IC50 = 296 nM T19368 CD50KP 90314195 IC50 = 19 nM T19368 CFIQ43 90314313 IC50 = 59 nM T19368 CAIX60 90315018 IC50 = 95 nM T19368 C0RX8W 90315177 IC50 = 19 nM T19368 CH48OX 90315197 IC50 = 25 nM T19368 C7JUT0 90330569 IC50 = 82 nM T19368 C3AF7K 90342616 IC50 = 61 nM T19368 CQ6RA9 117925769 IC50 = 1010 nM T19368 C64ROY 117926300 IC50 = 17 nM T19368 CJP74Z 117926496 IC50 = 231000 nM T19368 C4M3BV 117926681 IC50 = 32000 nM T19368 CT2D6S 117926717 IC50 = 48000 nM T19368 C6MCV9 117926750 IC50 = 50 nM T19368 CGC6I1 117926774 IC50 = 49 nM T19368 CNXE63 117926971 IC50 = 218 nM T19368 C9IES2 117927080 IC50 = 21 nM T19368 C7X1JK 117927107 IC50 = 156 nM T19368 C75MOW 118226885 IC50 = 4.6 nM T19368 C9YW2S 118226924 IC50 = 25 nM T19368 C0F9VX 118226926 IC50 = 7 nM T19368 CFI52X 118322776 IC50 = 90 nM T19368 CWU45F 118322800 IC50 = 1000 nM T19368 CQE12Y 118322815 IC50 = 200 nM T19368 C0YSJ1 118331270 IC50 < 10 nM T19368 C6RG9S 122681886 IC50 = 29 nM T19368 C5P4XN 132227197 IC50 = 13 nM T19368 C1R5SZ 132227201 IC50 = 50 nM T19368 C7NKD2 137375044 IC50 = 150 nM T19368 C1HPM0 138609421 IC50 = 130 nM T19368 C2EUS3 138609424 IC50 = 5.3 nM T19368 C98FIS 138609447 IC50 = 170 nM T19368 CN9B7C 138609489 IC50 = 1100 nM T19368 CCG37W 138609501 IC50 = 15 nM T19368 CRJ53U 138609502 IC50 = 16 nM T19368 C1U5QH 138632211 IC50 = 70 nM T19368 C0R2ZE 138632215 IC50 = 80 nM T19368 CG4RO6 138632227 IC50 = 30 nM T19368 CHT39X 138632268 IC50 = 50 nM T19368 CO4GV3 138632638 IC50 = 200 nM T19368 CVB6L2 138632650 IC50 = 30 nM T19368 CUQ3V8 155513144 IC50 = 7700 nM T19368 CKE03Y 155518423 IC50 = 20 nM T19368 C1LU5R 155527647 IC50 < 0.5 nM T19368 CA0L9Z 155527840 IC50 = 0.5 nM T19368 C6LH0P 155528700 IC50 = 450 nM T19368 C64HLU 155531285 IC50 < 0.5 nM T19368 C8GW4T 155535067 IC50 = 1 nM T19368 C28AOX 155536683 IC50 = 21 nM T19368 CGPM92 155537786 IC50 = 40 nM T19368 CBUK43 155559234 IC50 = 20 nM T19368 C85OCL 155561382 IC50 < 0.5 nM T19368 C27EOH 155563783 IC50 = 20 nM T19368 COM19F 155566437 IC50 = 2350 nM T19368 D0F1UD 4589192 IC50 = 100 nM T19368 D0L8ZG 79799 IC50 = 17000 nM T99954 D05ZTH 5311181 EC50 = 2.4 nM T99954 D06FEA 5280360 IC50 = 260 nM T99954 D0I4DQ 5280723 EC50 = 1.8 nM T99954 D0N2SR 9913767 EC50 = 6 nM T99954 D0WL5V 9867642 Ki = 6628 nM T99954 D00HTY 5280363 IC50 > 10000 nM T99954 D00IQH 11677589 Ki > 5000 nM T99954 D00MZK 9911469 Ki = 8.9 nM T99954 D03YAS 9824353 Ki > 10000 nM T99954 D08QWQ 5283081 EC50 > 10000 nM T99954 D0G6EI 9890801 Ki > 3200 nM T99954 D0GC5H 123879 IC50 > 100000 nM T99954 D0I3TU 45268455 IC50 > 100000 nM T99954 D0K1EG 11508736 IC50 > 10000 nM T99954 D0M4TJ 44219292 Ki = 3 nM T99954 D0RL4X 45270144 IC50 > 100000 nM T99954 D0X7EG 11462174 IC50 = 57900 nM T99954 D0W2OT 5311035 IC50 = 37 nM T99954 D02RUO 9807448 Ki > 10000 nM T99954 D08QHS 11296282 IC50 = 14414 nM T99954 D0G2XM 9847589 IC50 = 150 nM T99954 D0K0VH 9867949 IC50 > 10000 nM T99954 C53VYH 131814 IC50 = 160 nM T99954 CLM8P6 2114670 Ki > 25000 nM T99954 CX3LJ8 5283086 EC50 = 260 nM T99954 C2XLU7 5311228 Ki = 10000 nM T99954 CO7N1Z 5311239 IC50 > 10000 nM T99954 CC9BE3 6443852 EC50 = 26 nM T99954 C6TA3N 9809136 Ki = 21000 nM T99954 CV24TI 9817292 Ki > 76000 nM T99954 C58ADG 9823958 IC50 = 210 nM T99954 C64ZFW 9846782 Ki > 10000 nM T99954 C64QHP 9867899 Ki > 10000 nM T99954 CKMW12 9874010 Ki = 52000 nM T99954 C83ZAU 9886718 Ki > 10000 nM T99954 CF0HC5 9888589 IC50 > 10000 nM T99954 CFC8G4 9894720 Ki > 3000 nM T99954 CA5N0K 9895436 Ki = 21000 nM T99954 CKXD73 9910141 Ki > 10000 nM T99954 CKNG97 9931891 EC50 = 22 nM T99954 CQ1PM0 9934864 IC50 = 81 nM T99954 CICE70 9938626 Ki = 28300 nM T99954 CWDT69 9939791 Ki = 13000 nM T99954 C6SGH7 9954562 Ki > 500 nM T99954 C0BA3W 9955130 IC50 = 10 nM T99954 CYHR10 9955518 IC50 = 40 nM T99954 C4UK2Q 9955802 Ki = 610 nM T99954 CMPT81 10025456 IC50 > 10000 nM T99954 CQ3GW6 10047541 IC50 > 10000 nM T99954 C2I9SU 10090048 IC50 = 160 nM T99954 CVWO07 10090958 IC50 = 350 nM T99954 CNE21V 10095268 IC50 < 3162.28 nM T99954 CHF3N2 10095633 IC50 = 150 nM T99954 CEX2R1 10116114 Ki = 37 nM T99954 C73CXR 10116116 Ki = 200 nM T99954 C5Z3WL 10117702 Ki = 98 nM T99954 CH6K4Y 10139183 Ki = 2500 nM T99954 C8RZS5 10163305 Ki = 210 nM T99954 CEM21G 10181606 Ki = 7300 nM T99954 CY5K2P 10185382 Ki = 1000 nM T99954 C7Z2NA 10185612 Ki = 49 nM T99954 CW1B3U 10227894 Ki = 72 nM T99954 CW94KD 10228100 Ki = 320 nM T99954 C0ED9Y 10251023 IC50 > 10000 nM T99954 C8J9EN 10277744 Ki = 1100 nM T99954 CZN2K6 10278907 Ki = 92 nM T99954 CL7YG3 10287121 Ki > 13000 nM T99954 CQJI35 10299717 Ki = 130 nM T99954 C4CI1H 10300616 Ki = 430 nM T99954 CNT29F 10300724 Ki = 130 nM T99954 CRD7N8 10320441 IC50 = 650 nM T99954 CV8F7P 10321522 IC50 = 8 nM T99954 CFI8A5 10363130 Ki > 10000 nM T99954 CGK4N7 10367369 Ki > 10000 nM T99954 CB19MW 10402929 Ki = 37000 nM T99954 CNQS75 10410111 Ki > 10000 nM T99954 CLZ75P 10452166 IC50 = 700 nM T99954 CI1E3P 10477567 IC50 = 3100 nM T99954 C4K1TO 10477568 IC50 = 3000 nM T99954 CYTV60 10502508 IC50 > 10000 nM T99954 C39BYU 10502610 IC50 = 8900 nM T99954 CZ2H8E 10529261 IC50 > 10000 nM T99954 C4F9MA 10529683 IC50 = 3400 nM T99954 CANM20 10547489 IC50 > 10000 nM T99954 CTY02L 10552450 IC50 > 10000 nM T99954 C58ZOU 10552612 IC50 > 10000 nM T99954 C0D7EI 10553794 IC50 = 4500 nM T99954 CMO37F 10594576 IC50 > 10000 nM T99954 C3GKS1 10595288 IC50 > 10000 nM T99954 CJ7IT3 10599289 IC50 > 10000 nM T99954 CMY4P3 10601359 IC50 = 5900 nM T99954 CPV7D6 10623568 IC50 = 5000 nM T99954 CD13GN 10648014 IC50 > 10000 nM T99954 CI5HA0 10648334 IC50 > 10000 nM T99954 C9YQG5 10670992 IC50 > 10000 nM T99954 C9SUW2 10671942 IC50 = 1500 nM T99954 CP1Z8W 10694649 IC50 = 1400 nM T99954 C3WRM7 10696132 IC50 > 10000 nM T99954 C7H8NA 10717385 IC50 = 3300 nM T99954 C7GY6X 10739351 IC50 > 10000 nM T99954 CY8IB2 10740699 IC50 > 10000 nM T99954 C12SBH 10741017 IC50 > 10000 nM T99954 CG17HE 10741197 IC50 > 10000 nM T99954 CK8O4Z 10741899 IC50 > 10000 nM T99954 C64MLE 10767455 IC50 > 10000 nM T99954 CD1YX8 10813802 IC50 = 7500 nM T99954 CKST02 11122314 IC50 > 10000 nM T99954 C7H3LX 11166017 Ki = 680 nM T99954 CS1T9C 11174065 Ki = 630.96 nM T99954 CQ2IO4 11175906 Ki = 79.43 nM T99954 CO5T2P 11178659 Ki > 10000 nM T99954 CX3T0K 11186023 Ki = 251.19 nM T99954 C8G2JL 11186079 Ki = 79.43 nM T99954 C5BWJ0 11198334 Ki = 158.49 nM T99954 CF0M3A 11201307 Ki = 570 nM T99954 C61PSW 11201693 Ki = 400 nM T99954 C71EZB 11202310 Ki > 10000 nM T99954 CU7NJ3 11202399 Ki > 10000 nM T99954 CQB0I7 11208785 Ki = 398.11 nM T99954 C5VIH3 11220357 Ki = 251.19 nM T99954 COL08E 11224239 Ki = 6400 nM T99954 C4U0NF 11230941 Ki = 1000 nM T99954 C46IJM 11236846 Ki = 2600 nM T99954 C12OPV 11237257 Ki = 1900 nM T99954 CY07ZR 11243628 Ki = 79.43 nM T99954 CJU6I7 11244046 Ki = 501.19 nM T99954 C1X5HY 11244380 Ki = 794.33 nM T99954 C4S5MX 11249458 Ki > 10000 nM T99954 CZ87VH 11254374 Ki = 3162.28 nM T99954 CH6KT3 11255468 Ki = 316.23 nM T99954 CT6H2O 11259714 Ki > 10000 nM T99954 CLG1V9 11260449 Ki = 1800 nM T99954 C0LNI5 11260506 Ki = 3400 nM T99954 C6ZOS1 11261579 Ki = 530 nM T99954 CZ6X3N 11267409 Ki = 630.96 nM T99954 C70ESM 11269563 Ki = 14000 nM T99954 CR1QV7 11278428 Ki = 39.81 nM T99954 C8Y5TV 11282319 Ki = 750 nM T99954 CQ2V3R 11282605 Ki = 2900 nM T99954 CJ2V7N 11292620 Ki = 4700 nM T99954 CZU2D7 11293771 Ki = 560 nM T99954 C9E4SW 11294166 Ki > 20000 nM T99954 CA6C9B 11294449 Ki = 5200 nM T99954 C60SAH 11316066 Ki = 410 nM T99954 C8D5JF 11318288 Ki = 760 nM T99954 C2IJB0 11324024 Ki = 3981.07 nM T99954 CNT5Q2 11328662 Ki > 10000 nM T99954 C1PQ5Y 11336395 Ki = 31.62 nM T99954 CY96IG 11336790 Ki = 50.12 nM T99954 C4GC1Y 11350967 Ki = 270 nM T99954 CEU68T 11352417 Ki = 3500 nM T99954 CP8L6Q 11364260 Ki > 2300 nM T99954 CT0HN9 11370857 Ki = 630.96 nM T99954 CMEF37 11374771 Ki > 10000 nM T99954 CTHZ75 11374965 Ki = 210 nM T99954 CUZ19G 11375038 Ki > 10000 nM T99954 C3EJ7K 11381211 Ki = 630.96 nM T99954 CN2TG7 11387144 Ki > 3000 nM T99954 CND1W5 11390143 Ki < 10000 nM T99954 C0REY8 11391560 Ki = 794.33 nM T99954 C0THZ6 11392403 Ki = 50.12 nM T99954 C0QZH4 11402676 Ki = 1258.93 nM T99954 C2ED7O 11403716 Ki = 501.19 nM T99954 C9C4AG 11404217 Ki = 63.1 nM T99954 CWHO39 11407826 Ki = 80 nM T99954 CXPO04 11408533 Ki > 20000 nM T99954 C0SLC1 11409320 Ki > 10000 nM T99954 C4V0DU 11414893 Ki = 100 nM T99954 C8DVC5 11415742 Ki < 10000 nM T99954 C4NJ1R 11415934 Ki < 10000 nM T99954 CRJD01 11427479 Ki < 10000 nM T99954 C9VAG4 11431240 Ki > 10000 nM T99954 CUB3R5 11454655 Ki = 5800 nM T99954 CY1U4I 11460304 Ki = 316.23 nM T99954 C4PA6U 11460734 Ki = 5011.87 nM T99954 CE7RJ1 11460765 Ki = 3981.07 nM T99954 C6OR7L 11461526 Ki = 398.11 nM T99954 CVR8W9 11461588 Ki = 1258.93 nM T99954 CSE6D9 11465472 Ki > 10000 nM T99954 CJE7S9 11473193 Ki = 630.96 nM T99954 CZ4K0P 11476788 Ki > 21200 nM T99954 CE2JA4 11488860 Ki = 15510 nM T99954 C1W2ZK 11577792 Ki > 6000 nM T99954 C7Y6XJ 11597294 Ki = 400 nM T99954 C3BSV4 11696697 Ki > 13000 nM T99954 C9FPO5 11737623 Ki < 10000 nM T99954 CK60GP 11737656 Ki = 158.49 nM T99954 CS73JN 11739220 Ki = 50.12 nM T99954 CNYK74 11743212 Ki = 710 nM T99954 C8E4PV 11750835 Ki = 580 nM T99954 CX5R1A 11770925 Ki < 10000 nM T99954 C8V7NZ 11771014 Ki = 10000 nM T99954 CT34LO 13230981 Ki > 13000 nM T99954 CZ3TG0 13231966 Ki = 870 nM T99954 CO19GA 14372497 Ki > 2000 nM T99954 CB1N7G 14429703 EC50 > 10000 nM T99954 C9PVF4 15236833 IC50 = 18 nM T99954 C7F8CG 15290482 IC50 = 380 nM T99954 CQH2F8 15290495 IC50 = 8000 nM T99954 C87JKP 15290515 IC50 = 5300 nM T99954 C3JT1D 15428700 IC50 = 3900 nM T99954 C06OGJ 15486805 IC50 > 10000 nM T99954 C0L3VU 15486806 IC50 > 10000 nM T99954 CWQ8B9 15551228 Ki > 500 nM T99954 CT3R2K 15725728 IC50 > 10000 nM T99954 C20TAN 15725731 IC50 > 10000 nM T99954 CIS83K 15947857 Ki = 2000 nM T99954 C3L0RK 15948325 Ki > 7000 nM T99954 CK4FJ8 16664733 IC50 = 16 nM T99954 C76AIN 19377530 IC50 > 10000 nM T99954 CX08BC 21198692 Ki > 500 nM T99954 CHBP89 21877027 Ki = 25.12 nM T99954 CF51NZ 21893828 Ki = 5100 nM T99954 COPL52 22024188 Ki = 3162.28 nM T99954 CZO48L 22024191 Ki < 10000 nM T99954 C8KVW9 23355418 IC50 = 20 nM T99954 CF81SW 23582412 IC50 > 10000 nM T99954 CP2S4J 23663736 Ki = 6.1 nM T99954 CASU54 23696973 IC50 > 1000 nM T99954 C42LYP 24765153 Ki > 25700 nM T99954 CF72YI 24765671 Ki >= 785 nM T99954 C31JZP 24765672 Ki >= 2500 nM T99954 C4QX7Y 24765675 Ki >= 930 nM T99954 CL7Z9U 24765768 Ki >= 110 nM T99954 CT2W4R 24901436 IC50 = 77 nM T99954 CVXE16 24901437 IC50 = 66 nM T99954 CA2IJ7 24901438 IC50 = 138 nM T99954 CFE4O6 24901439 IC50 = 278 nM T99954 CSOV98 24901440 IC50 = 2133 nM T99954 CX31GO 24901441 IC50 = 358 nM T99954 CRJ26K 24901442 IC50 = 53 nM T99954 C5GU8F 24901443 IC50 = 296 nM T99954 CO3WK5 24901444 IC50 = 831 nM T99954 C1SLP4 24901445 IC50 = 1005 nM T99954 C8SV1K 24901446 IC50 = 741 nM T99954 CUOF95 24901447 IC50 = 4710 nM T99954 CY19MU 24901448 IC50 = 3480 nM T99954 COKH17 24901449 IC50 = 12200 nM T99954 C35CIF 24901451 IC50 = 3306 nM T99954 CFQA40 24952577 Ki > 7282 nM T99954 CD98IN 24952580 Ki > 456 nM T99954 C81WVN 24952927 Ki > 5474 nM T99954 CZT83E 24952928 Ki > 501 nM T99954 C8YHX3 24953283 Ki > 224 nM T99954 CZ93FO 24953285 Ki > 628 nM T99954 C17JTY 24953286 Ki > 2226 nM T99954 CFT0W5 24953624 Ki > 4992 nM T99954 C42VMD 24953625 Ki > 3461 nM T99954 C7B2EW 24953628 Ki > 2117 nM T99954 CXQJ67 25002382 Ki >= 1291 nM T99954 CN5SH9 25003075 Ki > 21000 nM T99954 CNOF71 44138108 Ki > 25700 nM T99954 CSRV98 44157014 IC50 = 1880 nM T99954 CHI65U 44159530 IC50 = 56200 nM T99954 CMNH53 44159772 IC50 = 33000 nM T99954 C2AV1K 44190762 IC50 = 6340 nM T99954 C0A4TB 44232564 EC50 = 18.5 nM T99954 C46VMC 44232565 EC50 = 7.8 nM T99954 CUL10P 44232568 EC50 = 23 nM T99954 CTK9I3 44233521 EC50 = 41 nM T99954 CJY6T1 44234028 Ki = 400 nM T99954 CQ13MH 44234032 Ki = 7 nM T99954 C5D2AV 44234532 EC50 = 21 nM T99954 C6B7YM 44234782 EC50 = 12 nM T99954 CVL8A5 44235044 EC50 = 3.3 nM T99954 CMG1Y5 44235291 EC50 = 19 nM T99954 CVBY63 44235519 EC50 = 3.9 nM T99954 CMJ1G3 44235520 EC50 = 6.6 nM T99954 CS5CZ3 44235521 EC50 = 3.4 nM T99954 C9T5SL 44235522 EC50 = 38 nM T99954 CM3L2H 44235755 EC50 = 10 nM T99954 CY76GT 44236221 EC50 = 5.2 nM T99954 C5RNO7 44266308 Ki = 316.23 nM T99954 CSOF28 44266708 IC50 = 23000 nM T99954 C1AGY0 44266710 IC50 = 7800 nM T99954 CS8P5L 44266736 IC50 = 4900 nM T99954 CN15JD 44266758 IC50 = 5300 nM T99954 CIS85L 44266768 IC50 = 600 nM T99954 CO09CG 44266775 IC50 = 9600 nM T99954 C8VHX5 44267032 IC50 = 220 nM T99954 CY3K7T 44267033 IC50 = 2100 nM T99954 C3X7HN 44267058 IC50 = 2200 nM T99954 CBM90L 44267196 IC50 = 460 nM T99954 CIB06W 44267244 IC50 = 2400 nM T99954 C76KNG 44267245 IC50 = 4200 nM T99954 C6BMG3 44267380 IC50 = 2000 nM T99954 CN90FE 44269464 Ki > 13000 nM T99954 C1L0ET 44269468 Ki > 13000 nM T99954 C5KRQ4 44269486 Ki > 13000 nM T99954 CL6M2P 44269516 Ki > 13000 nM T99954 CON8R9 44269520 Ki > 13000 nM T99954 C6MBG0 44269521 Ki > 13000 nM T99954 CZ3Q1L 44269523 Ki > 13000 nM T99954 CRL61O 44269532 Ki > 13000 nM T99954 C1Z4LU 44269540 Ki > 13000 nM T99954 CM72FA 44269542 Ki > 13000 nM T99954 CN0JV2 44269543 Ki > 13000 nM T99954 C28UJH 44269544 Ki > 13000 nM T99954 CR1IY6 44269568 Ki > 13000 nM T99954 CI3C9O 44269596 Ki > 13000 nM T99954 CC0EW9 44269597 Ki > 13000 nM T99954 CO5Q2A 44303590 Ki > 10000 nM T99954 CT95YO 44303626 Ki > 10000 nM T99954 C79VSM 44303627 Ki > 10000 nM T99954 C5UN6W 44303709 Ki > 10000 nM T99954 C10VUL 44303710 Ki > 10000 nM T99954 CI1M5F 44303711 Ki > 10000 nM T99954 C2IN1Z 44303723 Ki > 10000 nM T99954 C25ANM 44303889 Ki > 0.0001 nM T99954 C7PA9J 44303952 Ki > 10000 nM T99954 C2KJ4D 44303967 Ki > 0.0001 nM T99954 CD31HF 44303980 EC50 = 37 nM T99954 C9LUE1 44304008 Ki > 10000 nM T99954 CM15YG 44304009 Ki > 10000 nM T99954 CBV9D0 44304011 Ki > 10000 nM T99954 CVX8Y2 44304034 Ki > 10000 nM T99954 C10MFJ 44304051 Ki > 10000 nM T99954 C8VQ0P 44304052 Ki > 10000 nM T99954 CR29LI 44304055 Ki > 10000 nM T99954 C3D7QU 44304057 Ki > 10000 nM T99954 C9KN6Z 44304058 Ki = 510 nM T99954 C16ZGY 44304124 Ki > 10000 nM T99954 C9PM3Q 44304164 Ki > 10000 nM T99954 C2V9XR 44304181 EC50 = 25 nM T99954 CPB9V7 44304199 Ki > 0.0001 nM T99954 C86SPE 44304258 Ki > 10000 nM T99954 CW5X7C 44304334 Ki = 1400 nM T99954 C4IF3W 44304335 Ki > 10000 nM T99954 C94XIK 44304388 Ki = 750 nM T99954 CJ98YA 44304389 Ki > 10000 nM T99954 C5EWB3 44304403 Ki > 10000 nM T99954 CNA7I3 44304404 Ki > 10000 nM T99954 CT3QO5 44304417 Ki > 10000 nM T99954 CGN15F 44304436 Ki = 3.3 nM T99954 CV17WX 44304474 Ki = 920 nM T99954 CYQ29I 44326792 Ki = 80 nM T99954 CCG6V3 44344457 IC50 > 10000 nM T99954 C97ZYT 44356353 IC50 = 533 nM T99954 CLN63A 44377464 Ki = 31000 nM T99954 C5DV8H 44399137 Ki = 41 nM T99954 CRFL02 44400189 Ki = 170 nM T99954 CWL1X4 44400355 Ki > 1000 nM T99954 C76QVA 44402710 Ki = 140 nM T99954 CRAX23 44402824 Ki = 110 nM T99954 C3O4WY 44416263 IC50 = 115 nM T99954 CS5QJ2 44416265 IC50 = 114 nM T99954 CH21BU 44416278 IC50 = 53 nM T99954 CTY23X 44416280 IC50 = 39 nM T99954 CPC7W4 44416292 IC50 = 48 nM T99954 CZ1MD0 44416293 IC50 = 58 nM T99954 C3YCT7 44416333 IC50 = 930 nM T99954 CIB2W5 44419347 Ki > 500 nM T99954 C91JXT 44419374 Ki > 500 nM T99954 CNF4W2 44419379 Ki > 500 nM T99954 CYX21Z 44432434 IC50 = 3584 nM T99954 CDBE16 44450497 Ki > 22498 nM T99954 C6XE0K 44564841 IC50 > 10000 nM T99954 C0NF1S 44565193 IC50 = 4100 nM T99954 CQIK27 44627395 IC50 = 5875 nM T99954 C4W1ZG 44627515 IC50 = 8823 nM T99954 CULJ91 45268456 IC50 > 100000 nM T99954 CB5O6V 45269307 IC50 > 100000 nM T99954 C03ETI 45270148 IC50 > 100000 nM T99954 CY70SI 45270983 IC50 > 100000 nM T99954 C2XH3A 45270987 IC50 > 100000 nM T99954 C35DUQ 45272700 IC50 > 100000 nM T99954 CKUI32 45272704 IC50 > 100000 nM T99954 C3U7KT 45273637 IC50 > 100000 nM T99954 CS4F0X 46879894 IC50 > 20000 nM T99954 C2FR7X 46885690 IC50 > 20000 nM T99954 CN8D5V 46885691 IC50 > 20000 nM T99954 C9RP0X 46885735 IC50 > 20000 nM T99954 C0A2CI 46890616 Ki >= 504 nM T99954 CW52VH 46890658 Ki >= 260 nM T99954 CXQ2W0 46890659 Ki >= 580 nM T99954 CQ20RC 46890660 Ki >= 100 nM T99954 CM06FG 50898361 Ki > 7700 nM T99954 CZ9UD6 50901657 IC50 > 100000 nM T99954 CZ9D6X 53358921 Ki = 2200 nM T99954 COFI65 53358922 Ki = 200 nM T99954 CY40UL 53494965 Ki = 2600 nM T99954 CGC46Y 54764763 Ki > 10000 nM T99954 CQD5E9 56657974 Ki > 10000 nM T99954 CJV8Q3 56658143 Ki = 4600 nM T99954 C8OPY9 56658144 Ki > 10000 nM T99954 CC06JQ 56661509 Ki = 320 nM T99954 CX9UE6 56661510 Ki = 3000 nM T99954 C3LJ0H 56661652 Ki = 2700 nM T99954 CS65CK 56664920 Ki = 570 nM T99954 C4XP0K 56664921 Ki = 280 nM T99954 CR4U7M 56665068 Ki = 1600 nM T99954 CWR1Z7 56665984 Ki > 13000 nM T99954 C4PKJ5 56668353 Ki = 160 nM T99954 C4RN0E 56668527 Ki = 2900 nM T99954 C9DE7A 56671851 Ki = 2100 nM T99954 CWDP40 56672018 Ki > 10000 nM T99954 C4AOU2 56672019 Ki = 3500 nM T99954 C4ZE6P 56672020 Ki > 10000 nM T99954 CVF9P7 56675229 Ki = 91 nM T99954 CH3R8E 56675398 Ki = 3600 nM T99954 C73WGP 56675399 Ki = 1800 nM T99954 C9E3QR 56675400 Ki > 10000 nM T99954 CH3FS9 56678559 Ki = 94 nM T99954 CHN32S 56678560 Ki = 1500 nM T99954 C54DNU 56678561 Ki = 230 nM T99954 CMIX78 56681885 Ki = 110 nM T99954 CRQW04 56681898 Ki = 93 nM T99954 CM2BI9 56681899 Ki = 520 nM T99954 COE89W 56682059 Ki = 1400 nM T99954 C2MX5W 57391065 Ki = 3300 nM T99954 CC4UT1 57391066 Ki = 1700 nM T99954 C4FAZ8 57394587 Ki > 10000 nM T99954 CX4N6G 57396336 Ki > 10000 nM T99954 CQK50D 57401554 Ki = 520 nM T99954 CYG57I 57403305 Ki = 3300 nM T99954 C12SIB 58172125 EC50 = 25 nM T99954 C9MQ4Z 58602756 IC50 = 13 nM T99954 CI0A9L 68747456 EC50 > 10000 nM T99954 C6IHR3 68747472 EC50 > 10000 nM T99954 C5NZO0 68747479 EC50 > 10000 nM T99954 C8MED0 68749474 EC50 > 10000 nM T99954 CIUR89 68751402 EC50 > 10000 nM T99954 C8WC4E 68785185 EC50 = 2000 nM T99954 CJ7AY6 69753740 EC50 = 47 nM T99954 CQ9H4U 86277844 IC50 = 1000 nM T99954 CSJ4A9 118352160 EC50 = 4900 nM T99954 CE6L8I 118352177 EC50 > 10000 nM T99954 C8PKA7 118352211 EC50 > 10000 nM T99954 CPS7M4 118352285 EC50 = 5300 nM T99954 CLZJ36 118727285 EC50 = 969 nM T99954 CIM4J2 118727286 EC50 = 2670 nM T99954 CXWZ41 118727287 EC50 = 60 nM T99954 CL4AI3 118727288 EC50 = 180 nM T99954 CMDL48 118727289 EC50 = 380 nM T99954 C6X5EG 118727290 EC50 = 60 nM T99954 CB3QD7 118727291 EC50 = 37 nM T99954 CTC5J6 118727292 EC50 = 1720 nM T99954 CZ1S8B 118727293 EC50 = 1060 nM T99954 CGFH47 118727294 EC50 = 8.5 nM T99954 CKU5Z9 118727295 EC50 = 24 nM T99954 C9F1HX 118727296 EC50 = 114 nM T99954 CF6I8O 118727297 EC50 = 20 nM T99954 CE9G2Y 118727298 EC50 = 10 nM T99954 CCG76Q 118727299 EC50 = 9.5 nM T99954 CK9BJ0 118727300 EC50 = 62 nM T99954 CGAB46 118727301 EC50 = 100 nM T99954 CBN3D0 118727302 EC50 = 140 nM T99954 CVG17M 118727303 EC50 = 60 nM T99954 CQK7M2 118727304 EC50 = 86 nM T99954 CJ96RI 118727305 EC50 = 1060 nM T99954 CZNC59 118727306 EC50 = 120 nM T99954 C8HZ9I 118727307 EC50 = 38 nM T99954 C3IXH8 118727308 EC50 = 10 nM T99954 CPY2G0 118727309 EC50 = 140 nM T99954 C4E5GY 118727310 EC50 = 260 nM T99954 CJ0B3K 118727311 EC50 = 20 nM T99954 C0UP8I 118727312 EC50 = 4 nM T99954 C6DVX3 118727313 EC50 = 85 nM T99954 CEK5C9 118727314 EC50 = 33 nM T99954 C3L5VY 118727315 EC50 = 6 nM T99954 C9M4YO 118727316 EC50 = 79 nM T99954 C8ZRJ0 126495398 EC50 > 10000 nM T99954 C8SRZ5 126495427 EC50 > 10000 nM T99954 CD72CT 126495432 EC50 > 10000 nM T99954 CN72WL 126495463 EC50 > 10000 nM T99954 CV1A6C 126495491 EC50 > 10000 nM T99954 CYP3E5 126495507 EC50 = 1700 nM T99954 CPQU08 127028520 IC50 > 30000 nM T99954 CPN46Z 127028521 IC50 = 20000 nM T99954 C8D6KE 127028522 IC50 > 30000 nM T99954 CA9M1J 127028547 IC50 > 1000 nM T99954 C0ZCA9 127028548 IC50 > 1000 nM T99954 CW3HK5 127028549 IC50 > 1000 nM T99954 CNK1C6 127028550 IC50 > 1000 nM T99954 CU52FC 127028837 IC50 = 740 nM T99954 CI7Y2M 127028838 IC50 = 320 nM T99954 CLK95U 127028839 IC50 = 440 nM T99954 CGW85A 127028866 IC50 > 1000 nM T99954 CZ2LR3 127028867 IC50 > 1000 nM T99954 CQRL40 127029146 IC50 = 23000 nM T99954 CX9M6D 127029402 EC50 = 7900 nM T99954 C3QYS5 127029416 IC50 = 3200 nM T99954 CWXR72 127029417 IC50 = 130 nM T99954 CLB35Q 127029418 IC50 = 900 nM T99954 CK2E0B 127029419 IC50 > 1000 nM T99954 C0OIK8 127029420 IC50 = 430 nM T99954 CI4AN3 127029421 IC50 = 1000 nM T99954 CW1O4F 127029692 EC50 > 10000 nM T99954 CJAQ90 127047381 Ki = 400 nM T99954 CTR62O 127052613 EC50 = 11 nM T99954 CGZR45 127052614 EC50 = 2500 nM T99954 COVY75 127052615 EC50 > 10000 nM T99954 C4U3XA 134138103 EC50 > 10000 nM T99954 C10OQL 134144861 EC50 > 10000 nM T99954 CG0SO1 134147356 EC50 > 10000 nM T99954 C8QT5L 134149776 EC50 > 10000 nM T99954 C16HYX 134151657 EC50 > 10000 nM T99954 CIA76T 134157766 EC50 > 10000 nM T99954 CK5FQ9 137636847 EC50 = 1050 nM T99954 CGP4Z6 155544367 IC50 = 12500 nM T99954 D02MXT 24952929 Ki > 22000 nM T99954 D03OYD 5311240 IC50 > 10000 nM T99954 D05TNX 5311100 EC50 > 10000 nM T99954 D07UDT 15551229 Ki > 500 nM T99954 D08MNO 25886893 IC50 = 25 nM T99954 D0J9PG 119461 Ki > 100000 nM T99954 D0O9ES 5311053 IC50 > 10000 nM T99954 D0S2LO 9864831 Ki > 13000 nM T99954 D0TA0L 23685469 Ki = 54 nM T99954 D0Y1IF 23664784 Ki = 12 nM T99954 D0Z3XJ 9817405 Ki > 500 nM T44919 C41AIU 11169089 IC50 = 5000 nM T44919 CG43XJ 11376210 IC50 = 5000 nM T44919 CP56DO 11599295 IC50 = 6800 nM T44919 C6F4EX 44561438 IC50 = 5900 nM T44919 CSB74O 44561439 IC50 = 7600 nM T44919 C9Y2NP 44561556 IC50 = 3700 nM T06031 D02UFQ 11620908 IC50 > 10000 nM T06031 D04AHQ 71721540 IC50 = 98 nM T06031 D0E3TC 44259 IC50 = 485 nM T06031 D0O6ZO 9952773 IC50 > 10000 nM T06031 C0V7UW 9958506 IC50 > 11000 nM T06031 C1AKH9 10303277 IC50 = 8 nM T06031 C6FGQ1 25206346 IC50 > 10000 nM T06031 CU9E4P 42629114 IC50 = 8100 nM T06031 CEL61X 44229839 IC50 > 10000 nM T06031 C3VRO9 44557921 IC50 > 10000 nM T06031 C6E2SC 45482700 IC50 > 10000 nM T06031 CZXH74 45482750 IC50 > 10000 nM T06031 CUA97D 46209401 IC50 > 10000 nM T06031 CT3EW2 59292007 IC50 > 1000 nM T06031 CV63UL 67240318 IC50 > 10000 nM T06031 CEBO91 71452977 IC50 > 10000 nM T06031 CHQZ25 71459584 IC50 > 10000 nM T06031 CZ31PU 71583657 IC50 > 10000 nM T06031 C86HPW 155518524 IC50 = 66000 nM T65116 D0F2XQ 657237 Ki = 500000 nM T65116 CDJ4K6 5987 IC50 = 42100 nM T65116 C7MHL3 7009 IC50 = 21800 nM T65116 C7N9ZC 7022 IC50 = 1320 nM T65116 C2MU7H 8479 IC50 = 8200 nM T65116 CRT69E 70070 Ki = 2000000 nM T65116 C41OCL 174223 IC50 = 13500 nM T65116 C4V8YB 193201 Ki = 4.57 nM T65116 CR5PJ0 9889639 IC50 = 2000 nM T65116 C64FOA 13742375 IC50 = 41000 nM T65116 CV51PK 16067130 Ki = 1000000 nM T65116 CL82ST 19967710 IC50 = 30500 nM T65116 CB5QW4 76324498 IC50 = 47600 nM T65116 CTBL86 91669228 Ki = 893300 nM T65116 CM75YG 122185397 Ki = 4.51 nM T65116 C4EBU3 126672948 IC50 > 1000000 nM T65116 CP2F6A 127047463 Ki = 64 nM T65116 CQJT80 127047464 Ki = 138 nM T65116 C0GLP7 127047465 Ki = 46 nM T65116 C5XZT3 127047466 Ki = 42 nM T65116 C3QVE9 127047481 Ki = 18 nM T65116 C96CIU 127047596 Ki = 338 nM T65116 CZJ73D 127047597 Ki = 18 nM T65116 CPHO79 127047598 Ki = 91 nM T65116 C3W6MA 127047642 Ki = 63 nM T65116 C9ZAE0 127047727 Ki = 79 nM T65116 CI3X7G 127047728 Ki = 27 nM T65116 CI95SW 127047759 Ki = 53 nM T65116 CZP84Q 127048134 Ki = 14 nM T65116 C0RO4M 129217302 IC50 = 3162.28 nM T65116 CCO1S6 129229125 IC50 = 15.85 nM T65116 CK0FV5 130205852 Ki = 0.005 nM T65116 CI20GW 130205896 IC50 = 2200 nM T65116 C5Z6PW 130206267 IC50 = 180 nM T65116 C7T2WK 135406506 Ki = 255 nM T65116 C1D4FC 145925611 Ki = 35.7 nM T65116 CFA36V 145925613 Ki = 15.4 nM T65116 CZ2YD3 145925614 Ki = 184 nM T65116 CQ57LX 145961953 IC50 = 63.1 nM T65116 C9L0ZW 145962755 IC50 <= 316.23 nM T65116 CB8Q2X 145962960 IC50 = 1000 nM T65116 CTFP35 145963579 IC50 = 100 nM T65116 C6QO4S 145996542 Ki = 3.33 nM T65116 CAU3Z1 146020618 IC50 = 18.9 nM T65116 C2ZQ5W 146020619 IC50 = 220 nM T65116 CS54CM 146433251 IC50 = 49.5 nM T65116 CGO5C4 146433253 IC50 = 12.4 nM T65116 CJ15FL 146433266 IC50 = 9200 nM T65116 C5RYZ7 146433270 IC50 = 5100 nM T65116 CMWU18 146433315 IC50 = 306 nM T65116 CB7Y0L 146433462 IC50 = 333 nM T65116 C61LGO 146433463 IC50 = 63.1 nM T65116 CQ7LO1 146433473 IC50 = 21 nM T65116 C4OSN5 146433538 IC50 = 56 nM T65116 CN2MA4 146433574 IC50 = 56.5 nM T65116 CMH2X4 146676950 Ki = 0.318 nM T65116 CKN9I4 153538536 IC50 = 1030 nM T65116 CE4GO2 155511330 IC50 = 12000 nM T65116 C5NHY9 155511705 IC50 = 22300 nM T65116 CZH0J4 155511748 IC50 = 10000 nM T65116 CUR12T 155511776 IC50 = 6750 nM T65116 COD1Y3 155513204 IC50 = 12400 nM T65116 C32KPT 155515482 IC50 > 1000000 nM T65116 CZ3D8K 155515689 IC50 > 1000000 nM T65116 C0SR9Q 155516147 IC50 = 2390 nM T65116 C84ZUF 155516372 Ki = 6.29 nM T65116 C5LUP8 155516521 Ki = 7.96 nM T65116 C4LMN7 155516730 IC50 = 142 nM T65116 CKVA67 155517112 IC50 = 651 nM T65116 CUH12R 155519853 IC50 > 1000000 nM T65116 CU5TL6 155520896 IC50 = 54400 nM T65116 CRQ7Y1 155521443 IC50 = 141 nM T65116 C5TK1O 155522801 IC50 = 68100 nM T65116 C1OCJ2 155523491 IC50 = 78 nM T65116 CO5ZE9 155523514 IC50 = 140000 nM T65116 CYI71L 155523951 IC50 = 46.1 nM T65116 C65NJS 155524405 IC50 = 5200 nM T65116 CYU02N 155524529 Ki = 23.6 nM T65116 C1TQ9S 155524688 IC50 > 1000000 nM T65116 C2MAS4 155524869 IC50 = 49000 nM T65116 CY7V9B 155525421 IC50 = 148000 nM T65116 C8AO2P 155525981 IC50 = 331 nM T65116 CE8C1U 155526109 IC50 = 5350 nM T65116 C4OD7G 155526114 IC50 = 97300 nM T65116 CYTV51 155526138 IC50 > 1000000 nM T65116 CQ0P3W 155526883 IC50 > 1000000 nM T65116 CZ94CG 155527952 IC50 > 1000000 nM T65116 CQ9C6U 155529949 IC50 = 54 nM T65116 CFY6I9 155531322 IC50 = 480 nM T65116 CP98GU 155533987 IC50 = 162 nM T65116 C59WCH 155534198 IC50 = 9000 nM T65116 C65UWS 155534564 Ki = 15.9 nM T65116 C2PZV1 155534704 IC50 = 1100 nM T65116 CJ3P5W 155534768 IC50 = 121000 nM T65116 CRS63L 155535046 IC50 = 594 nM T65116 C3TN0U 155535612 IC50 > 1000000 nM T65116 C9T8ZV 155535856 IC50 = 1700 nM T65116 CM6T4Q 155535967 Ki = 61.9 nM T65116 C4ZYC0 155536729 IC50 = 210 nM T65116 CJWV24 155537635 IC50 > 1000000 nM T65116 CW54VO 155538959 IC50 = 15610 nM T65116 CVJT14 155539753 IC50 > 1000000 nM T65116 CB43YR 155540395 IC50 = 53.5 nM T65116 CAX9G3 155540458 IC50 > 1000000 nM T65116 CT83QU 155540535 Ki = 4.58 nM T65116 CA8RP3 155541438 Ki = 842700 nM T65116 CNH46F 155543687 IC50 = 54.7 nM T65116 C3FJ0I 155544707 IC50 = 2850 nM T65116 CYO2K8 155545063 IC50 = 65 nM T65116 CK45XL 155545753 IC50 = 3690 nM T65116 CP16WE 155547856 IC50 > 1000000 nM T65116 C7Z4UF 155548302 IC50 = 178500 nM T65116 C5EG0K 155548570 Ki = 46.9 nM T65116 C9K0JV 155549025 IC50 > 1000000 nM T65116 CDA51K 155550469 IC50 = 45 nM T65116 C0XTV2 155552570 IC50 > 1000000 nM T65116 CR0G4F 155553249 IC50 = 646 nM T65116 C5JYT2 155553286 IC50 = 224 nM T65116 C9N3DE 155553296 IC50 = 14200 nM T65116 CSXF92 155553772 IC50 > 1000000 nM T65116 C3SGB2 155555897 Ki = 10.1 nM T65116 C6T3NB 155556423 IC50 = 47000 nM T65116 CBIY07 155557730 IC50 > 1000000 nM T65116 CJZ9M8 155561535 IC50 = 408 nM T65116 C1MW3L 155561646 IC50 = 57 nM T65116 C0Q2YU 155562134 IC50 = 99000 nM T65116 CP39KL 155563743 IC50 > 1000000 nM T65116 CR3UO0 155563848 IC50 = 13700 nM T65116 CLA0W8 155564699 IC50 > 1000000 nM T65116 CDIK04 155565046 IC50 > 450000 nM T65116 C90WKD 155565469 IC50 > 1000000 nM T65116 CNT16A 155566608 IC50 > 1000000 nM T65116 CBVE71 155567059 IC50 = 9000 nM T65116 CG0JH2 155567373 IC50 = 360 nM T65116 CEV3T5 155567875 IC50 = 191000 nM T65116 CFR7B8 155568365 IC50 = 269 nM T65116 D0O9GJ 92199 Ki = 88.4 nM T68668 CW96BH 446222 Ki = 1430000 nM T68668 C62ZHS 10331137 Ki = 152470 nM T68668 CL2K5P 10932483 Ki = 332950 nM T68668 CQFD27 10988011 Ki = 232800 nM T68668 CHUK42 11126680 Ki = 1310000 nM T68668 CO0U4R 11277122 Ki = 35980 nM T68668 CFE5J4 11290388 Ki = 7770 nM T68668 C6Q4FY 11414083 Ki = 29880 nM T68668 C1KS4Z 11416597 Ki = 68270 nM T68668 CPQ02T 11425273 Ki = 26930 nM T68668 C24CON 11484266 Ki = 25900 nM T68668 CLDB75 11485203 Ki = 9140 nM T68668 C4ZTF8 11737619 Ki = 11800 nM T68668 C59WNV 13329882 Ki = 530610 nM T68668 CSM95J 16104237 Ki = 4350 nM T68668 CYT8A7 45093274 Ki = 567640 nM T68668 C86EXR 45093275 Ki = 292020 nM T68668 CPQ49A 71450639 Ki = 43150 nM T68668 CVR0H8 71452507 Ki = 64910 nM T68668 C4S0MT 71454231 Ki = 437720 nM T68668 CD2F4N 71454232 Ki = 15480 nM T68668 C0N2AM 71455988 Ki = 11270 nM T68668 C35MHZ 71457787 Ki = 6470 nM T68668 CA0KM1 71457788 Ki = 12810 nM T68668 CCO96R 71457789 Ki = 450360 nM T68668 CMN41F 71457830 Ki = 80850 nM T68668 CB78SH 71459708 Ki = 683000 nM T68668 CXV0T4 71459737 Ki = 82350 nM T68668 C0FLT2 71459738 Ki = 123030 nM T68668 CW0VG7 71461463 Ki = 229380 nM T89534 D00ZFP 5870 EC50 = 0.7 nM T89534 D01XBA 5035 Ki = 0.03 nM T89534 D06LOQ 179337 EC50 = 0.2 nM T89534 D06NXY 5991 IC50 = 2 nM T89534 D06XMU 6013 IC50 > 10000 nM T89534 D07BSQ 5994 IC50 > 1000 nM T89534 D07KSG 2733526 IC50 = 8 nM T89534 D08QMX 5757 EC50 = 0.004 nM T89534 D09NMD 216416 IC50 = 1.3 nM T89534 D0D1SG 5755 Ki > 5000 nM T89534 D0EP0C 5833 Ki > 1100 nM T89534 D0JO7Y 104741 IC50 = 0.06 nM T89534 D0JY8T 154257 IC50 = 3.7 nM T89534 D0Q4SD 443872 IC50 > 10000 nM T89534 D0V9BD 2375 Ki > 100000 nM T89534 D0X1EZ 2898 EC50 = 26 nM T89534 D0Y2NE 448537 EC50 = 0.007 nM T89534 D0Y7IU 5281004 IC50 > 10000 nM T89534 D0Y7JU 9854489 IC50 > 5000 nM T89534 D0Z1FX 5756 EC50 = 1.995 nM T89534 D0Z4EI 55245 Ki > 200 nM T89534 D00JFE 56941241 Ki = 0.37 nM T89534 D01SYU 10026128 IC50 = 10000 nM T89534 D07LZH 656954 IC50 = 1216 nM T89534 D09NST 449459 IC50 = 0.79 nM T89534 D0L4FS 5280961 IC50 = 9.7 nM T89534 D0LI1C 44469321 IC50 > 30000 nM T89534 D0R2SK 10286159 Ki = 2.29 nM T89534 D0SZ1G 121248172 IC50 > 100000 nM T89534 D0TN6K 118574930 IC50 = 6 nM T89534 D0U3EP 445154 Ki = 785 nM T89534 D0X1OW 86287635 IC50 = 0.138 nM T89534 D0X9YP 67041274 IC50 > 10000 nM T89534 D02KAU 46871935 IC50 > 10000 nM T89534 D03KTE 16750192 Ki > 10000 nM T89534 D05BCA 68570 EC50 = 1.5 nM T89534 D08DZZ 10634 EC50 = 26 nM T89534 D08HIH 6102691 IC50 = 210 nM T89534 D09AAM 104772 IC50 = 50 nM T89534 D09UFV 24825740 IC50 > 10000 nM T89534 D0H5CV 130936 IC50 = 25 nM T89534 D0J4ZH 3033898 Ki = 46.29 nM T89534 D0R8TB 6433099 EC50 = 0.1 nM T89534 D0U7OU 3220 Ki = 770 nM T89534 D0W5RL 9577221 IC50 = 1900 nM T89534 CXMH37 6620 IC50 = 133 nM T89534 C3EUZ1 6776 Ki = 310 nM T89534 C8GBH5 7184 IC50 = 1420 nM T89534 C6QYD8 8434 EC50 = 38200 nM T89534 CHA7C3 12111 EC50 = 909 nM T89534 CVUW13 14128 IC50 = 8970 nM T89534 CGWM38 54900 IC50 = 0.72 nM T89534 CSI62C 62082 EC50 = 6.5 nM T89534 CQ0IC4 63062 Ki = 0.04 nM T89534 CH98UA 65511 IC50 = 34600 nM T89534 CF5JU9 75386 IC50 = 230 nM T89534 CYCI69 80152 EC50 = 75.1 nM T89534 CNT0H1 96201 IC50 = 170 nM T89534 CS8Q6W 99649 Ki = 5700 nM T89534 CMEN50 101689 IC50 > 5000000 nM T89534 CM9CO5 119588 Ki = 41.5 nM T89534 C5E2IG 223998 Ki = 8 nM T89534 C78YGO 232446 IC50 = 520 nM T89534 C8MJB2 247310 IC50 = 84 nM T89534 CDHI70 251929 IC50 = 640 nM T89534 C9XC2A 252281 IC50 > 10000 nM T89534 CDP78A 261349 EC50 = 540 nM T89534 CZJW92 348148 EC50 = 80 nM T89534 C7HME8 439246 IC50 = 75302 nM T89534 CKB57V 440624 IC50 = 11000 nM T89534 C5SEF1 442342 IC50 1000000 nM T89534 C40YBS 444036 IC50 > 10000 nM T89534 CJZO27 445920 Ki = 4.1 nM T89534 CK01NI 448577 IC50 = 0.8 nM T89534 CGT37O 449205 IC50 = 0.5 nM T89534 C9AXQ3 449207 IC50 = 0.4 nM T89534 CBD7O2 449208 IC50 = 1.3 nM T89534 CL26SB 449209 IC50 = 1.3 nM T89534 CMT3P0 480764 EC50 = 5 nM T89534 C5UM8B 513197 EC50 = 1400 nM T89534 C0CF9H 586500 IC50 = 85700 nM T89534 CZ0AH3 638278 IC50 = 1870 nM T89534 C9UW8R 640096 EC50 = 2030 nM T89534 C2I3PM 646429 IC50 = 2230 nM T89534 CB20EC 656952 IC50 = 46 nM T89534 C67LKM 656953 IC50 = 1152 nM T89534 C2KCS3 667696 EC50 = 800 nM T89534 C2B0JA 674359 Ki = 15000 nM T89534 CX8H6W 687290 IC50 = 7980 nM T89534 C3R1PZ 721251 IC50 = 2320 nM T89534 C1OG7J 833976 EC50 = 12800 nM T89534 CV95AN 837745 IC50 = 28200 nM T89534 C31BFY 837746 EC50 = 31100 nM T89534 C69DLW 837838 IC50 = 4320 nM T89534 C4T6YS 837853 IC50 = 28100 nM T89534 C06JQG 837872 IC50 = 3060 nM T89534 CQOD41 837886 IC50 = 1000 nM T89534 C1ZE2H 845978 IC50 = 290 nM T89534 C6XGH8 849252 IC50 = 1200 nM T89534 C9S4EA 849257 IC50 = 2290 nM T89534 CE9VY2 849282 IC50 = 430 nM T89534 C4IQG9 849291 IC50 = 629 nM T89534 CN6RA2 849298 IC50 = 1980 nM T89534 CPQ72T 849308 IC50 = 31600 nM T89534 C45RBT 851153 EC50 = 3080 nM T89534 CO85AF 902564 EC50 > 100000 nM T89534 C5MZH8 906479 IC50 1000000 nM T89534 C2LRG9 927532 EC50 = 203 nM T89534 C5A7CD 928630 IC50 1000000 nM T89534 C90CUZ 1111980 EC50 > 10000 nM T89534 C6YNU8 1131384 Ki > 10000 nM T89534 C23KHO 1132609 IC50 < 100000 nM T89534 C5GJF1 1234611 IC50 = 3150 nM T89534 CM6NY1 1234663 IC50 = 1890 nM T89534 CMBE67 1234708 IC50 = 3290 nM T89534 C7TE0L 1717570 EC50 = 18700 nM T89534 CF4S1M 1731992 IC50 = 8770 nM T89534 C8WS4M 2040507 IC50 1000000 nM T89534 CLF0C9 2288503 IC50 = 24 nM T89534 CS6TF7 2733525 IC50 = 1700 nM T89534 C6LXG3 2747677 IC50 = 74 nM T89534 CFH19O 2887782 IC50 = 1100 nM T89534 CBZ6U1 3024714 IC50 = 285 nM T89534 C5GVH1 3035198 IC50 = 4 nM T89534 C7RNA9 3325226 IC50 = 16.48 nM T89534 C0F8EP 3519901 EC50 = 400 nM T89534 C9S2LO 4055843 EC50 = 4130 nM T89534 C6J0ZF 4369568 IC50 = 1.5 nM T89534 CFY94M 4369569 IC50 = 0.8 nM T89534 CL9G3U 4608762 EC50 > 10000 nM T89534 CH6RY7 5282240 EC50 = 11.2 nM T89534 CB6OK2 5287464 IC50 = 24 nM T89534 C7IBX9 5287551 IC50 = 8 nM T89534 CJB7T6 5288494 IC50 < 3.2 nM T89534 CW91XD 5322257 EC50 = 43.8 nM T89534 CS31LU 5322291 EC50 = 231 nM T89534 CP69KZ 5324349 EC50 = 21.4 nM T89534 C2JOL1 5327043 Ki = 0.47 nM T89534 CN7CS6 5372367 IC50 = 61.91 nM T89534 CF5VB6 5395460 IC50 1000000 nM T89534 C9GS2K 5397219 EC50 = 59.1 nM T89534 CQ83GI 5397398 IC50 1000000 nM T89534 C4Z1IB 5400235 EC50 = 331 nM T89534 CNG5W4 5407968 IC50 > 10000 nM T89534 CO36YU 5455071 EC50 = 35800 nM T89534 C52EHD 5822393 IC50 = 4660 nM T89534 CY9MR6 5885714 IC50 = 2320 nM T89534 CT0F6H 5948122 IC50 = 120 nM T89534 C6LCX3 6260040 EC50 = 415 nM T89534 CL41HW 6303362 EC50 = 95 nM T89534 C16ZSG 6439929 IC50 = 62000 nM T89534 C6RDY2 6444422 EC50 = 0.52 nM T89534 C3E0BP 6604873 EC50 = 2.9 nM T89534 C1VLY9 6918261 IC50 = 0.04 nM T89534 CF61LI 7314046 IC50 = 255 nM T89534 CM5Y0Z 7314049 IC50 = 795 nM T89534 CXHO01 7314090 IC50 = 10800 nM T89534 CFM7Q8 7314234 IC50 = 2870 nM T89534 C3M7RE 9804246 IC50 = 31 nM T89534 CU3QR8 9808162 Ki = 120 nM T89534 CNJE78 9811391 IC50 = 80 nM T89534 CE23GX 9814262 IC50 = 624 nM T89534 C34IZS 9814547 IC50 = 114 nM T89534 CZA2O0 9814673 EC50 = 794 nM T89534 CCUR98 9815144 IC50 = 344 nM T89534 CTB3F6 9815173 IC50 = 24 nM T89534 C4C7HN 9816479 IC50 > 200000 nM T89534 CNJK98 9816989 Ki = 10 nM T89534 CX1F7P 9819159 IC50 = 122.7 nM T89534 CTXR52 9820272 EC50 > 100000 nM T89534 CT78HP 9823190 IC50 > 10000 nM T89534 CN9M3P 9824019 Ki = 0.9 nM T89534 C94INP 9829162 IC50 = 2430 nM T89534 C7V2ZD 9835427 IC50 = 1650 nM T89534 CCX60E 9835779 IC50 = 1050 nM T89534 CHE70V 9838722 Ki > 100000 nM T89534 CS97CD 9846731 IC50 = 1 nM T89534 C2LV3C 9848252 IC50 = 1 nM T89534 CMI0N6 9848501 Ki = 0.32 nM T89534 CQGZ49 9856356 EC50 > 1000 nM T89534 CVW25C 9856632 EC50 = 671 nM T89534 C8ER6V 9869745 Ki = 210 nM T89534 C9MA0B 9878811 EC50 = 59 nM T89534 CIA6K1 9878841 EC50 = 460 nM T89534 CJ8VH6 9879228 IC50 = 5982 nM T89534 CPF25S 9879409 IC50 = 2420 nM T89534 CA1CJ6 9879798 IC50 = 273 nM T89534 C01ZFV 9882789 IC50 > 10000 nM T89534 CIT93X 9884138 IC50 = 141 nM T89534 CL8E7Z 9890509 IC50 = 0.7 nM T89534 CL7UB1 9900112 IC50 = 195 nM T89534 C3EQA8 9900383 EC50 = 449 nM T89534 C30BCU 9900479 IC50 = 264 nM T89534 CM9S2I 9900695 IC50 = 883 nM T89534 C3C6GN 9902151 IC50 = 41 nM T89534 C2BUL1 9902785 EC50 = 561 nM T89534 C38PGE 9903336 IC50 = 9.5 nM T89534 CB63ZP 9907598 IC50 = 500 nM T89534 CLC48G 9909681 IC50 = 0.5 nM T89534 CCZ9P8 9911175 Ki > 10000 nM T89534 CD3A6G 9912022 Ki = 0.6 nM T89534 C6YGM0 9912245 IC50 = 3 nM T89534 C58PVC 9921352 IC50 = 455 nM T89534 CJL2P9 9921784 IC50 = 976 nM T89534 CBX75P 9922298 IC50 = 30 nM T89534 CGN5C8 9922681 EC50 = 681 nM T89534 CX9AV7 9923647 EC50 = 1267 nM T89534 CJD4H0 9923941 IC50 = 70.5 nM T89534 CFT7M0 9924049 IC50 = 19 nM T89534 C9I3SQ 9924986 IC50 = 1410 nM T89534 CE6HU3 9925763 Ki = 4.34 nM T89534 CP8ZG3 9927355 Ki = 11 nM T89534 C39EXP 9933936 IC50 = 2281 nM T89534 CVW4Y8 9935633 IC50 = 7.8 nM T89534 CB0H3V 9942858 IC50 = 1210 nM T89534 CB65XA 9943599 IC50 > 10000 nM T89534 CW4RV2 9945087 EC50 = 1178 nM T89534 CO4IM2 9946131 IC50 = 663 nM T89534 C81CGQ 9946229 EC50 = 870 nM T89534 CZP05L 9948127 Ki = 3.3 nM T89534 CQ04ES 9948426 IC50 > 10000 nM T89534 CY6M2H 9953602 IC50 = 10.69 nM T89534 C9OPU4 9957008 Ki = 160 nM T89534 CEK90Y 9958368 Ki = 3.9 nM T89534 CO5V0P 9964601 IC50 = 1190 nM T89534 C0AJ3H 9964943 EC50 = 1233 nM T89534 CJT98P 9965271 IC50 = 630 nM T89534 C0LGC8 9965955 EC50 = 120 nM T89534 C1ZBV6 9967036 IC50 = 128 nM T89534 C29KIM 9968828 EC50 = 94 nM T89534 C4XGS5 9970588 Ki = 4 nM T89534 C05NAQ 9973567 IC50 = 597 nM T89534 CKS02X 9974556 EC50 = 620 nM T89534 COJ0E4 9993475 IC50 = 228 nM T89534 C4V6RF 9998996 IC50 > 1000 nM T89534 CB6AC7 10002045 IC50 = 1.4 nM T89534 CDU28H 10005346 IC50 = 2 nM T89534 CW4B6F 10015172 IC50 = 3074 nM T89534 CJN7T4 10016716 IC50 = 4160 nM T89534 C3XCR4 10016731 IC50 = 129 nM T89534 C7NLS3 10016946 IC50 = 7485 nM T89534 C8UT2P 10019713 IC50 = 4258 nM T89534 CG8B1H 10026593 IC50 = 1.6 nM T89534 CE0X1Y 10038212 IC50 = 1580 nM T89534 C0XGJ2 10043907 EC50 = 65 nM T89534 C3QBA5 10060912 IC50 = 14300 nM T89534 C9Z0AT 10060945 IC50 = 159 nM T89534 CUCM03 10062125 Ki > 100000 nM T89534 CIY1Z7 10064013 IC50 = 2521 nM T89534 C37ZQE 10072011 Ki = 8.69 nM T89534 C8P1BZ 10084254 IC50 = 3030 nM T89534 CDM8V3 10084479 IC50 = 716 nM T89534 CT1ZO9 10085265 IC50 = 33248 nM T89534 CYH2U5 10086047 IC50 = 627 nM T89534 CMDP60 10107798 IC50 > 10000 nM T89534 CM4B3Q 10108320 IC50 = 1160 nM T89534 C96JZH 10113416 IC50 = 4.7 nM T89534 C4XU7H 10115709 IC50 = 1 nM T89534 C9EDV6 10115710 IC50 = 0.8 nM T89534 CCA85G 10125282 IC50 = 55 nM T89534 CWLS93 10125319 IC50 = 1402 nM T89534 CTF5J0 10125414 Ki = 0.35 nM T89534 CH4N0B 10125582 IC50 = 356 nM T89534 CYIT90 10125667 IC50 = 10 nM T89534 CRP1U3 10128287 IC50 = 0.7 nM T89534 C08BYF 10140504 IC50 = 0.7 nM T89534 CQK5X9 10144672 Ki = 475 nM T89534 CC24WL 10149300 IC50 > 5000 nM T89534 CO1AE6 10149393 IC50 = 1650 nM T89534 C8G4PV 10149522 IC50 = 10 nM T89534 CY15UJ 10149610 IC50 = 118 nM T89534 C2EOX1 10151898 IC50 = 0.61 nM T89534 CIEH85 10154586 EC50 = 49 nM T89534 C0MX7K 10157532 IC50 > 10000 nM T89534 C1BAI4 10171529 Ki = 40 nM T89534 CT5W0A 10171640 IC50 = 12 nM T89534 CD36GZ 10171641 IC50 = 3.1 nM T89534 C36ACW 10171666 IC50 = 143 nM T89534 C5I7DH 10171723 Ki = 2.88 nM T89534 C9P4CF 10171732 IC50 = 548 nM T89534 C5DSH0 10171830 IC50 = 125 nM T89534 C3QR7A 10171898 IC50 = 9 nM T89534 CK0ZU9 10172081 IC50 = 710 nM T89534 C1VDO4 10174471 IC50 = 3.8 nM T89534 CJO0M8 10174620 IC50 = 1.1 nM T89534 C2YRA6 10177915 IC50 = 124 nM T89534 C8L7HJ 10179031 IC50 > 10000 nM T89534 C2BS8L 10181886 Ki = 1.7 nM T89534 CWCM45 10182934 Ki = 0.6 nM T89534 C3JZH5 10183377 EC50 = 200 nM T89534 CKT6Z4 10183386 IC50 = 18 nM T89534 CQB51M 10184149 IC50 = 0.9 nM T89534 C0J9AT 10184212 IC50 = 5.2 nM T89534 CG5N8H 10184413 Ki = 490 nM T89534 C8XEP4 10192873 IC50 = 180 nM T89534 CR48FY 10192874 IC50 > 5000 nM T89534 CP70BT 10192899 IC50 = 21 nM T89534 C3RV4A 10192967 Ki = 41 nM T89534 CT19KI 10192968 Ki = 65 nM T89534 CVM71O 10192978 IC50 = 1056 nM T89534 CY3ZU9 10193027 IC50 = 114 nM T89534 C1UF6W 10193573 IC50 = 200 nM T89534 C73GTR 10204098 IC50 = 11.9 nM T89534 CS91YM 10210142 Ki = 675 nM T89534 CH02FU 10214626 IC50 = 6 nM T89534 C4PKF0 10214678 Ki = 267 nM T89534 CJN2Y4 10214684 IC50 > 5000 nM T89534 CP90ZM 10214912 IC50 = 480 nM T89534 C82SVD 10215058 IC50 = 299 nM T89534 C8GZN0 10215089 IC50 = 5.2 nM T89534 CP4U5C 10215240 IC50 = 47 nM T89534 CP41MR 10215241 IC50 = 3 nM T89534 C7PSG6 10215290 IC50 = 21 nM T89534 C0FU1V 10215342 IC50 = 131 nM T89534 CP1S2V 10217796 IC50 = 4 nM T89534 CU2RI4 10217951 IC50 = 1 nM T89534 CW05OU 10218853 IC50 > 10000 nM T89534 CJ9BE0 10222329 IC50 > 10000 nM T89534 C84SRT 10223610 IC50 > 10000 nM T89534 CGF4E7 10226687 IC50 = 3 nM T89534 C7FXG9 10227720 IC50 = 172 nM T89534 C5M1RH 10229852 Ki = 360 nM T89534 CNB84J 10236378 IC50 = 2951 nM T89534 CVMD95 10236407 IC50 = 58 nM T89534 CV9SZ3 10236450 IC50 = 109 nM T89534 C1K8OP 10236507 IC50 = 2 nM T89534 C7CPB9 10238739 IC50 = 51 nM T89534 CMY87N 10243978 EC50 = 6.7 nM T89534 C7E0OP 10244111 IC50 = 488 nM T89534 C0JE2W 10248828 IC50 = 1440 nM T89534 CJQZ83 10254189 Ki = 0.5 nM T89534 CS4B5C 10265236 IC50 = 46 nM T89534 CPBH94 10266789 IC50 = 43 nM T89534 CGV0O2 10268080 IC50 = 196 nM T89534 CR59SC 10271193 IC50 > 10000 nM T89534 CPIS57 10271557 IC50 > 10000 nM T89534 CPZY03 10275313 Ki = 2.5 nM T89534 C7LHP1 10275916 Ki > 1000 nM T89534 CL5P3T 10276036 Ki = 120 nM T89534 CBD8V6 10282029 EC50 = 150 nM T89534 C7G4RE 10286186 IC50 = 40 nM T89534 C15UPR 10286213 IC50 = 40 nM T89534 C37GHD 10286369 IC50 = 35 nM T89534 C4U9ZV 10286370 IC50 = 519 nM T89534 CS4Y7Z 10286462 IC50 = 290 nM T89534 CUQC81 10287415 IC50 > 1000 nM T89534 CM8IW0 10288944 IC50 = 2.6 nM T89534 CLOE40 10291224 IC50 = 5880 nM T89534 C04JEC 10299557 IC50 = 110 nM T89534 C10CJA 10308134 IC50 = 105 nM T89534 CGR20A 10308169 IC50 = 31 nM T89534 C1KY6P 10308176 IC50 = 23 nM T89534 CX15KH 10308458 IC50 = 36 nM T89534 C7R4NE 10308501 Ki = 6.11 nM T89534 C0VUR6 10308538 IC50 = 580 nM T89534 COP14A 10312439 IC50 > 1000 nM T89534 COHA43 10316618 IC50 = 225 nM T89534 C1FLQ0 10323601 Ki = 34 nM T89534 CPJS68 10324755 Ki = 1.22 nM T89534 C5K2CL 10332429 IC50 > 10000 nM T89534 C7R6EP 10332721 IC50 = 1280 nM T89534 CO2IH4 10334049 IC50 = 4382 nM T89534 CPK7W1 10344612 Ki = 32 nM T89534 C0YAJ6 10344970 IC50 = 0.7 nM T89534 CEA16J 10344977 IC50 = 2.7 nM T89534 C1MH2K 10346077 EC50 = 1800 nM T89534 C35BTN 10355544 IC50 = 10000 nM T89534 CMY0N8 10355768 IC50 = 435 nM T89534 C61WZX 10356510 IC50 = 9830 nM T89534 C5YU0I 10358550 IC50 = 6850 nM T89534 CR98BH 10358677 IC50 = 1920 nM T89534 C7SO6W 10361788 IC50 = 9 nM T89534 CEJ78I 10365592 IC50 > 2000 nM T89534 CKD8I0 10370518 IC50 = 5 nM T89534 CBG59N 10377168 IC50 = 550 nM T89534 CGCE89 10378417 IC50 = 484 nM T89534 CRB41T 10379126 IC50 = 25956 nM T89534 C14AIB 10384345 IC50 > 2000 nM T89534 C6RQK1 10386584 IC50 > 10000 nM T89534 CYN9E1 10390108 EC50 = 200 nM T89534 CK8MI6 10390296 IC50 = 1.3 nM T89534 CH9P0A 10390835 IC50 = 61 nM T89534 CJV0O5 10400919 IC50 = 1780 nM T89534 C7JN6F 10401620 IC50 = 626 nM T89534 C40NPC 10407651 Ki > 100000 nM T89534 CQ46GH 10412249 Ki = 0.28 nM T89534 C1P4XA 10414598 IC50 = 5.6 nM T89534 CA80YJ 10423234 IC50 = 11097 nM T89534 C6H7EJ 10423780 IC50 = 10000 nM T89534 CPM1L8 10425817 IC50 = 11600 nM T89534 CC1V4Y 10428321 IC50 = 373 nM T89534 C98YGB 10430074 IC50 = 597 nM T89534 C04EKD 10436416 IC50 > 10000 nM T89534 C8ZS3V 10447061 IC50 > 6260 nM T89534 CZ08NR 10447944 IC50 = 29.8 nM T89534 CH58OG 10450569 EC50 = 15 nM T89534 C0NT9D 10454007 IC50 > 5000 nM T89534 CM92LK 10467580 IC50 = 583 nM T89534 C4JK0T 10468337 IC50 = 785 nM T89534 CLV49C 10470279 EC50 = 243 nM T89534 C6UMY7 10471178 IC50 = 3120 nM T89534 CB8PK9 10473796 EC50 = 1740 nM T89534 C85RBN 10474264 IC50 > 2000 nM T89534 CUL8O4 10475384 IC50 > 1000 nM T89534 CMG35I 10478373 IC50 = 2.5 nM T89534 C8GZN6 10479379 IC50 = 1.9 nM T89534 CZB0G1 10480448 IC50 = 65 nM T89534 CAL8E3 10719917 IC50 = 0.046 nM T89534 CM69RP 10768122 Ki = 0.25 nM T89534 CC7N5G 10809406 IC50 > 11 nM T89534 C30MWO 10812923 EC50 = 1660 nM T89534 CC2L7D 10814352 IC50 < 0.002 nM T89534 C39FWK 10858337 EC50 = 40 nM T89534 CKTE95 10863480 Ki > 10000 nM T89534 CT1L6K 10874604 Ki > 10000 nM T89534 C2W9QX 10885394 IC50 = 71 nM T89534 C75IVW 10892270 EC50 = 464 nM T89534 C4ZI0B 10897174 Ki > 10000 nM T89534 CNZ9H2 10901682 EC50 = 191 nM T89534 CMW1U8 10906531 Ki = 1420 nM T89534 CJP54O 10906754 Ki = 200 nM T89534 CY5R8D 10908233 Ki = 1050 nM T89534 C40LHE 10917513 Ki > 10000 nM T89534 C3WI4P 10917876 IC50 = 46 nM T89534 CJ8OD1 10923143 EC50 = 18 nM T89534 CU46XG 10928571 IC50 = 2.9 nM T89534 CS24AP 10928882 IC50 = 3.097 nM T89534 COM46T 10929139 Ki = 145 nM T89534 CJ3RF6 10930298 Ki = 1300 nM T89534 C3HG2S 10933614 EC50 = 178 nM T89534 C5E8VA 10938971 Ki = 5130 nM T89534 CK5D4I 10939453 IC50 = 0.6998 nM T89534 CT8B7X 10940598 Ki = 180 nM T89534 C1OQB3 10945098 EC50 = 71200 nM T89534 CH14AY 10950078 Ki = 6870 nM T89534 CJL36T 10950356 Ki > 10000 nM T89534 CZ8F4V 10950649 IC50 = 2.897 nM T89534 CP2IK4 10950883 IC50 = 4.498 nM T89534 C3I5PB 10952341 Ki = 1450 nM T89534 C4VD3H 10955612 EC50 = 3.1 nM T89534 CR94QD 10956181 EC50 = 148 nM T89534 CD90TL 10961334 Ki = 2400 nM T89534 CZGP46 10967017 EC50 = 16 nM T89534 CI9PC0 10972569 EC50 = 500 nM T89534 C7KSR9 10972765 Ki = 570 nM T89534 CW7ND8 10973721 Ki = 6320 nM T89534 CW52ES 10973841 Ki = 810 nM T89534 CC4UT6 10978897 EC50 = 2.9 nM T89534 C93KBD 10978965 EC50 > 1000 nM T89534 CF2WJ3 10983822 Ki = 560 nM T89534 C2Q9UC 10985075 Ki = 855 nM T89534 C79JBL 10993930 IC50 = 2.6 nM T89534 CL1I0Z 10994057 Ki = 290 nM T89534 CW62AM 10999188 EC50 = 269 nM T89534 C1N8ZM 10999677 EC50 = 48 nM T89534 CGSE70 11011115 EC50 = 2.7 nM T89534 CE4C5I 11015765 IC50 = 2.999 nM T89534 CWO8S9 11016369 Ki = 1000 nM T89534 CHR7A9 11016735 Ki = 125 nM T89534 CG37VC 11022432 EC50 = 162 nM T89534 CH9Y1B 11026647 IC50 = 0.5998 nM T89534 CGX1N0 11028495 Ki = 1130 nM T89534 COE9W8 11037182 Ki = 2370 nM T89534 CZW72E 11037591 IC50 = 3.5 nM T89534 C3JH4N 11039284 Ki = 2040 nM T89534 CNG30Q 11048590 Ki > 10000 nM T89534 C2Z6TH 11048839 Ki = 415 nM T89534 CQN16G 11048858 IC50 = 3.3 nM T89534 C5W9IK 11060085 Ki = 2275 nM T89534 CWO84P 11060104 Ki = 830 nM T89534 CV1A6F 11070590 Ki = 1140 nM T89534 CF9LM6 11070635 Ki = 270 nM T89534 CU9PY6 11071460 EC50 = 180 nM T89534 CWG41U 11075979 EC50 = 23 nM T89534 C2L7DT 11086416 EC50 = 363 nM T89534 C09ZLY 11088436 Ki > 10000 nM T89534 CG3VQ7 11091722 IC50 = 1.5 nM T89534 C8ED0O 11092497 Ki = 480 nM T89534 C49GHR 11097061 EC50 = 0.38 nM T89534 CX8YU9 11102748 IC50 = 44 nM T89534 CD1G4U 11102972 Ki = 570 nM T89534 CR8OQ5 11114635 Ki = 2360 nM T89534 CDJW25 11117751 EC50 = 209 nM T89534 C1O8RD 11124781 Ki > 10000 nM T89534 CGH0S4 11135858 Ki = 570 nM T89534 CNEX86 11146178 Ki = 3000 nM T89534 CIG8Z6 11153316 Ki > 100000 nM T89534 CJ4S8B 11153461 EC50 > 10000 nM T89534 CJ12UZ 11155391 IC50 = 0.66 nM T89534 CS2B4Z 11155392 IC50 = 1.4 nM T89534 CJ7KZ9 11155655 Ki > 100000 nM T89534 CP7R9U 11156432 EC50 = 1700 nM T89534 C4SEB7 11160528 IC50 = 790 nM T89534 CGI4Y2 11162677 Ki > 1000 nM T89534 CT0JD9 11164713 EC50 > 1000 nM T89534 C5DM4H 11165305 IC50 = 38 nM T89534 C68FNC 11167858 IC50 = 1090 nM T89534 CX91QE 11185437 IC50 = 343 nM T89534 CVAI71 11186162 EC50 = 1000 nM T89534 CBS6E8 11197092 IC50 = 180 nM T89534 CAPL61 11197251 IC50 = 45 nM T89534 C9T6KS 11197891 Ki > 100000 nM T89534 CLQ9C4 11197931 Ki = 8.3 nM T89534 C1XPD4 11201600 IC50 = 18 nM T89534 CB1FI6 11201991 IC50 = 1.3 nM T89534 CO2N4Z 11208222 Ki > 100000 nM T89534 C0M4IP 11208678 Ki = 700 nM T89534 CN6V7O 11209303 Ki > 100000 nM T89534 CDG4Q2 11221797 EC50 > 10000 nM T89534 C3M5WN 11224950 IC50 = 2.4 nM T89534 CA7F5T 11225110 EC50 = 1500 nM T89534 C7M9AJ 11230651 Ki > 100000 nM T89534 CN27ZJ 11231364 IC50 = 73 nM T89534 C2Q5PJ 11231792 IC50 = 186 nM T89534 CMIO31 11235808 EC50 = 780 nM T89534 CQHW46 11243890 Ki > 100000 nM T89534 C3B4HX 11244016 Ki > 100000 nM T89534 C5IM4X 11247367 Ki = 1.7 nM T89534 C3RM9N 11254549 IC50 = 235 nM T89534 C5A7JR 11254851 IC50 = 406 nM T89534 CNJ4Q3 11255230 IC50 = 6324 nM T89534 CYCR06 11256303 IC50 > 10000 nM T89534 CWF3M2 11256602 Ki = 12.4 nM T89534 CEA6U1 11259746 IC50 = 5.1 nM T89534 CZ1LG3 11266077 Ki > 100000 nM T89534 CIRO56 11267448 IC50 = 64908.26 nM T89534 C7N9EL 11268331 IC50 = 116 nM T89534 CC0XI4 11279959 IC50 > 10000 nM T89534 C4SC0W 11281576 IC50 > 1000 nM T89534 C8LFT9 11287739 Ki > 100000 nM T89534 C69KHE 11294796 IC50 = 2.5 nM T89534 C5A1NL 11300439 IC50 = 96 nM T89534 CY2GB4 11300595 Ki = 380.8 nM T89534 CS5HC9 11300885 EC50 = 11 nM T89534 CI7CZ3 11301461 IC50 = 55 nM T89534 C0XUF2 11305564 IC50 > 5000 nM T89534 CP61NH 11310856 Ki > 100000 nM T89534 C8S5AR 11314096 Ki = 7.2 nM T89534 C5M2KX 11317852 IC50 = 0.7 nM T89534 COU8G6 11323885 IC50 = 434 nM T89534 C61YIJ 11326213 EC50 = 5000 nM T89534 C1HZS7 11336351 IC50 > 10000 nM T89534 CL0TH7 11338484 EC50 = 3470 nM T89534 C1ZJ2R 11338969 IC50 = 31 nM T89534 CH12WB 11339036 IC50 = 153 nM T89534 CT9Y4O 11339440 IC50 > 10000 nM T89534 CBN46V 11340868 Ki = 1.03 nM T89534 C2T7ZW 11350120 EC50 > 10000 nM T89534 CU6BE2 11350495 IC50 = 34.9 nM T89534 C6YUB4 11350836 IC50 = 38 nM T89534 CR1EB4 11351870 IC50 = 19.6 nM T89534 CSNT72 11357451 IC50 = 84 nM T89534 CW3L1T 11358876 Ki > 100000 nM T89534 C8Z3YW 11359856 Ki = 4.2 nM T89534 CT3WZ0 11361524 IC50 = 46.6 nM T89534 C8AW4J 11363477 IC50 = 1.3 nM T89534 C90MRZ 11368962 EC50 = 35 nM T89534 C1HS3D 11369558 IC50 = 113 nM T89534 CMSU02 11370317 Ki = 410 nM T89534 C68GMX 11375318 EC50 = 1820 nM T89534 CXO72T 11376166 EC50 = 85 nM T89534 CTL6Z7 11382252 EC50 = 3000 nM T89534 CEI5V6 11385564 IC50 = 119 nM T89534 CK42BA 11391793 IC50 = 247 nM T89534 CL8JI2 11391816 Ki > 100000 nM T89534 C8G2ED 11397112 IC50 = 1.6 nM T89534 C17SXG 11397412 IC50 = 0.5 nM T89534 CO15AK 11403179 IC50 = 73 nM T89534 CS6VA1 11406904 IC50 = 55 nM T89534 CUC6L8 11407390 IC50 = 87 nM T89534 C0L2IW 11414230 Ki > 100000 nM T89534 CYM9V2 11414783 Ki > 100000 nM T89534 CO20QH 11416730 IC50 > 10000 nM T89534 C9YW0P 11425113 Ki > 100000 nM T89534 CC9D7U 11427021 EC50 = 984 nM T89534 C5WO0U 11429662 IC50 > 1000 nM T89534 CM9VH4 11430588 IC50 = 63 nM T89534 CFXR09 11431084 EC50 = 500 nM T89534 CGF15N 11431657 IC50 = 177 nM T89534 C0VR7F 11437418 IC50 = 26 nM T89534 CP7J9V 11437506 IC50 = 231 nM T89534 CYIU98 11438491 Ki > 100000 nM T89534 C6QK5H 11441393 EC50 > 10000 nM T89534 C2NMY6 11465422 IC50 = 3 nM T89534 CFG6L2 11471499 IC50 = 527 nM T89534 C8B9ZT 11471500 IC50 = 254 nM T89534 CK75PT 11476995 IC50 = 2.84 nM T89534 CP4M8J 11482995 Ki = 136 nM T89534 CNUG46 11487991 IC50 = 1.5 nM T89534 C3PNE7 11493187 IC50 = 11111 nM T89534 C7D5BU 11493338 IC50 = 5365 nM T89534 CN3W8L 11493379 IC50 = 6200 nM T89534 CFPW12 11496802 Ki = 0.3 nM T89534 CM76FT 11496925 Ki = 1.89 nM T89534 CQZ37A 11515143 IC50 = 81324 nM T89534 C4OBS2 11517134 Ki = 692 nM T89534 C5W9CK 11517889 IC50 = 3.5 nM T89534 CJ2WY6 11522286 EC50 = 4.3 nM T89534 C9G5AE 11536973 EC50 = 494 nM T89534 C5W8HY 11537063 EC50 = 622 nM T89534 CMOL82 11540768 Ki = 0.57 nM T89534 CS0O5B 11554672 EC50 = 3100 nM T89534 CUK47O 11558075 IC50 = 15521 nM T89534 CWCZ35 11558237 IC50 = 13240 nM T89534 CR4D8K 11558528 EC50 = 982 nM T89534 CP9GR8 11561520 Ki = 2 nM T89534 CSF3D4 11565065 EC50 = 10600 nM T89534 CUD60X 11565235 IC50 = 9635 nM T89534 C5YO1V 11565733 IC50 = 55015 nM T89534 C7UDF3 11565847 IC50 = 10649 nM T89534 C19NWZ 11565922 EC50 = 344 nM T89534 CWOZ42 11572578 IC50 = 66860 nM T89534 C07ALM 11582925 IC50 = 14 nM T89534 CKV64Z 11582975 Ki = 28 nM T89534 C4IZK8 11587711 EC50 = 14 nM T89534 CGQ5M2 11587774 IC50 = 770 nM T89534 C29NKX 11597321 IC50 = 18000 nM T89534 C9QS7V 11605525 Ki = 5.8 nM T89534 C92NWX 11610210 IC50 = 5 nM T89534 CC21VD 11610867 Ki = 59 nM T89534 CNP72K 11615788 EC50 = 0.31 nM T89534 CA3ID6 11619024 Ki = 52 nM T89534 CB10RY 11623915 EC50 = 324 nM T89534 C8M6GX 11631082 EC50 = 47 nM T89534 C7PG3I 11633183 Ki = 60 nM T89534 C45XNL 11637913 IC50 = 43968 nM T89534 CQ8EI7 11638242 Ki = 0.67 nM T89534 C60DQS 11638602 EC50 = 603 nM T89534 CA7S2I 11644884 IC50 = 34626 nM T89534 C2MQE5 11644885 IC50 = 121 nM T89534 CD2TL1 11645057 EC50 = 158 nM T89534 C7NBT6 11645733 EC50 > 1000 nM T89534 CK7ZQ8 11647673 IC50 = 0.6 nM T89534 C9LZ1F 11651922 IC50 = 43814 nM T89534 C84GDU 11655056 IC50 = 13000 nM T89534 CI1E3R 11659178 EC50 = 0.059 nM T89534 C3GXI8 11659260 IC50 = 44175 nM T89534 C1QV8H 11660523 Ki = 198 nM T89534 CWL7S9 11662094 IC50 = 29000 nM T89534 C0LKN3 11663272 EC50 = 152 nM T89534 CF4HM7 11666535 IC50 = 19437 nM T89534 CX2W9Z 11666644 IC50 = 6247 nM T89534 CJ2UC4 11674336 IC50 = 101544 nM T89534 CB1DU8 11674420 EC50 = 17 nM T89534 C3IK0P 11680776 IC50 = 15297 nM T89534 CH7O4Y 11681405 IC50 = 178 nM T89534 CJL8A6 11681415 EC50 = 10 nM T89534 CFZ0K5 11688293 EC50 = 3.9 nM T89534 CZ35CY 11694886 IC50 = 70277 nM T89534 CQ0IP3 11695307 IC50 = 70399 nM T89534 C20PTC 11696330 Ki = 2.1 nM T89534 CC6VK8 11702683 EC50 = 719 nM T89534 C0FEB7 11710790 EC50 = 427 nM T89534 CG4E2O 11719093 Ki = 4 nM T89534 C43LND 11720175 Ki = 0.24 nM T89534 CRP5H6 11720774 EC50 = 100 nM T89534 CR52IJ 11722356 EC50 > 1000 nM T89534 C7D9HG 11724363 IC50 > 10000 nM T89534 CO3S2Z 11724477 IC50 = 10000 nM T89534 CWK56G 11730419 Ki = 1000 nM T89534 CBMR23 11730420 Ki > 10000 nM T89534 C4FXP3 11730578 Ki = 200 nM T89534 C4GDB9 11730602 IC50 = 5.2 nM T89534 CB8J4L 11730916 Ki = 60 nM T89534 C1I0ZW 11733031 Ki = 3240 nM T89534 CT40UX 11734564 Ki = 1025 nM T89534 CGZ40Y 11738040 IC50 = 312 nM T89534 C4DCI8 11738269 IC50 = 2329 nM T89534 C9I3LZ 11738605 EC50 = 344 nM T89534 CF0D1S 11740374 EC50 = 1860 nM T89534 CCT71E 11743602 Ki = 1380 nM T89534 C9KTN0 11744183 Ki = 1.1 nM T89534 C0K4LB 11749762 Ki = 49000 nM T89534 CEC20W 11750375 IC50 = 18.2 nM T89534 C5YF3X 11750707 IC50 = 162 nM T89534 C5JH1M 11751440 IC50 = 122 nM T89534 CA2DO6 11770898 IC50 = 98 nM T89534 CHX6E0 11776977 IC50 = 4590 nM T89534 CH7VT9 11777076 IC50 = 3710 nM T89534 CD4W6C 11777154 IC50 = 1860 nM T89534 C98FDE 11777375 EC50 = 138 nM T89534 CNLQ34 11777905 IC50 = 1000 nM T89534 CT8OB2 11777956 IC50 = 97982 nM T89534 CL76UG 11778912 EC50 > 1000 nM T89534 CS9K7Z 11812018 IC50 = 1.799 nM T89534 CS4X7T 11817441 Ki > 100000 nM T89534 C8YD5R 11823753 EC50 = 42 nM T89534 CYQ0W7 11826815 IC50 = 19 nM T89534 CUVE20 11826959 Ki = 680 nM T89534 CT6Z4P 11827881 Ki = 250 nM T89534 C2VDT9 11954121 IC50 = 5.9 nM T89534 CFB48H 11957006 IC50 = 793 nM T89534 C3F6JK 11977778 EC50 = 870 nM T89534 C2CXT4 11987846 IC50 = 129 nM T89534 CSK1Q4 12019124 IC50 > 5000 nM T89534 COR2Z7 12074176 Ki = 0.21 nM T89534 C2HNA8 12083341 IC50 = 2728 nM T89534 C4U8KY 12085089 IC50 > 10000 nM T89534 COZ0Q5 12085941 IC50 = 28.7 nM T89534 C0P4TJ 12085942 IC50 = 562 nM T89534 C06AOU 12117259 EC50 = 65 nM T89534 C0IJ4C 12130940 EC50 = 300 nM T89534 CD2K0P 12130943 EC50 = 150 nM T89534 C41TJX 12258274 IC50 = 3672 nM T89534 CTZ92I 12642771 IC50 = 39400 nM T89534 C5GV6L 13613337 IC50 = 2530 nM T89534 C1J0CU 13720325 EC50 = 4 nM T89534 CS38YQ 14065243 EC50 = 15 nM T89534 CK2O7U 14128123 EC50 = 1500 nM T89534 CTU56S 14496018 EC50 = 1200 nM T89534 C42MYO 15429026 IC50 = 10.9 nM T89534 CB7K0N 15521393 IC50 = 3.53 nM T89534 C9NSQ7 15542995 EC50 = 5 nM T89534 C9IUR6 15543000 IC50 = 94 nM T89534 C0Q5RP 15543001 EC50 = 13 nM T89534 CF0U2J 15543006 EC50 = 336 nM T89534 COW27A 15543007 EC50 = 28 nM T89534 CZB7P9 15543008 EC50 = 40 nM T89534 C8J6DM 15543009 IC50 = 3.5 nM T89534 C49NDP 15887827 EC50 = 10 nM T89534 CUO82C 15984114 EC50 = 10.4 nM T89534 C2CVH9 15984115 EC50 = 8.3 nM T89534 CWF0I6 16007239 EC50 = 519 nM T89534 CR2Q9N 16038396 Ki = 1700 nM T89534 CV4LD2 16082545 IC50 = 82 nM T89534 C7S4XY 16082546 IC50 = 440 nM T89534 CKGI59 16082547 IC50 = 5500 nM T89534 C5ZJR4 16082550 IC50 = 1200 nM T89534 CR8NQ7 16082556 IC50 = 22 nM T89534 CUOE19 16082557 EC50 = 14 nM T89534 CIWO01 16082558 EC50 = 11 nM T89534 CW2EC8 16082559 IC50 = 40 nM T89534 CZ3N1E 16082564 IC50 = 160 nM T89534 C9WS2L 16082565 IC50 = 140 nM T89534 COR9P3 16082566 EC50 = 300 nM T89534 CH8A7C 16082568 IC50 = 340 nM T89534 C9O5EM 16082572 IC50 = 14 nM T89534 CK7PI6 16082573 IC50 = 25 nM T89534 C9QXI4 16082574 IC50 = 25 nM T89534 C7GL5X 16082575 EC50 = 41 nM T89534 C2BOE6 16103238 Ki = 266 nM T89534 C4UFW5 16103245 Ki = 408 nM T89534 CKHS18 16106496 IC50 < 100000 nM T89534 C95OTV 16106497 IC50 < 100000 nM T89534 CT17EJ 16106503 IC50 < 100000 nM T89534 C6H0EQ 16655080 IC50 = 36 nM T89534 C1UY8J 16666386 IC50 > 5000 nM T89534 C1F5XE 16719760 IC50 = 666 nM T89534 CE6FQ8 16719863 IC50 = 35.6 nM T89534 C7N4LJ 16719865 Ki = 0.63 nM T89534 C0PMA8 16719866 IC50 = 19.3 nM T89534 CC82UX 16720250 IC50 = 27 nM T89534 CWK35C 16730429 IC50 = 29000 nM T89534 CM4BS9 16739367 IC50 = 2 nM T89534 CZ34MS 16750039 IC50 = 8 nM T89534 CVSA61 16750040 IC50 = 1 nM T89534 CQZK05 16758226 Ki = 43.8 nM T89534 C3M8BI 17010631 IC50 < 100000 nM T89534 CVBN30 17191222 IC50 = 44.43 nM T89534 CE4CP2 17756206 IC50 = 193 nM T89534 C2AP6N 17760561 EC50 = 2.6 nM T89534 C4DV6C 17964485 Ki = 88 nM T89534 C9B3MR 17972677 IC50 = 1990 nM T89534 C4UG6E 17972712 IC50 = 4410 nM T89534 C84OYE 18172398 IC50 = 4.7 nM T89534 CS1C5Q 18172400 IC50 = 30.7 nM T89534 C30ALH 18172403 IC50 = 165 nM T89534 CZ0VW4 18172409 IC50 = 385 nM T89534 C5U1YK 18172442 IC50 = 29.4 nM T89534 CJ05MC 18172444 IC50 = 42.7 nM T89534 CUS3Z9 18172448 IC50 = 160 nM T89534 C3X1FG 18172450 IC50 = 28 nM T89534 CTVK47 18172466 IC50 = 6.7 nM T89534 CR53UZ 18172469 IC50 = 24.8 nM T89534 C93MVX 18172476 IC50 = 9.2 nM T89534 CCE1L5 18172477 IC50 = 50 nM T89534 C0RZB8 18172482 IC50 = 235 nM T89534 C9DS4J 18695694 Ki = 2 nM T89534 CJ9RH8 19087421 IC50 > 200000 nM T89534 CGP29U 19793984 IC50 = 2900 nM T89534 C1F4KI 19793985 IC50 = 84 nM T89534 C95KIE 20160413 IC50 = 1.3 nM T89534 CI0P6T 20161167 IC50 = 14 nM T89534 CSY05K 20227298 IC50 = 1.3 nM T89534 CM86ZJ 20734982 IC50 = 3 nM T89534 C0Q4FT 21051956 IC50 = 0.28 nM T89534 CF0S6J 21210483 IC50 > 30000 nM T89534 CV2N4Y 21252247 EC50 = 72 nM T89534 C7WBV5 21355678 IC50 = 53.6 nM T89534 CUL35V 21433016 IC50 = 79 nM T89534 C0HG2O 21625144 EC50 > 10000 nM T89534 C4BON1 21628493 EC50 = 0.028 nM T89534 CY56XC 21868866 EC50 = 0.3 nM T89534 C0AVF8 21868918 IC50 = 3 nM T89534 C6MTN2 21959300 IC50 = 23 nM T89534 CQS75R 22064611 Ki = 29 nM T89534 C89GZT 22221606 IC50 = 625 nM T89534 C5R3ZU 22221614 IC50 = 263 nM T89534 CD52LR 22221618 IC50 = 103 nM T89534 CU3E0Q 22221630 IC50 = 109 nM T89534 CN94JH 22221634 IC50 = 49 nM T89534 CC6X3H 22600576 IC50 > 10000 nM T89534 CT8Q2E 23349396 IC50 = 115 nM T89534 C7W5VE 23424169 IC50 = 7980 nM T89534 C6TJY8 23509070 EC50 = 16.2 nM T89534 C9O6RB 23596322 Ki > 5000 nM T89534 C8FN7B 23648275 IC50 = 17.2 nM T89534 C4TNI0 23648457 Ki = 126 nM T89534 CZGS14 23648464 Ki = 2.82 nM T89534 CBL4I8 23648465 Ki = 27.2 nM T89534 CK0XL8 23648466 Ki = 147 nM T89534 C0GP7Q 23653178 IC50 = 2650 nM T89534 CV04HC 23653179 IC50 = 1630 nM T89534 CPR38W 24015539 EC50 = 5950 nM T89534 CTE1N2 24748569 EC50 > 10000 nM T89534 C4WYE7 24749678 Ki > 1100 nM T89534 C2QHO3 24749808 Ki > 1100 nM T89534 CP7M4B 24768258 EC50 = 1000 nM T89534 CH4QT2 24768259 EC50 > 1000 nM T89534 C8DS1F 24825443 IC50 = 100 nM T89534 CZ4P8I 24825444 IC50 = 200 nM T89534 C7PR1H 24825445 IC50 = 25 nM T89534 CZ9O3D 24825446 IC50 = 1 nM T89534 CW43SX 24825447 IC50 = 13 nM T89534 CKW98C 24825448 IC50 = 10 nM T89534 CN9TA0 24825453 IC50 = 250 nM T89534 CF1H9X 24825454 IC50 = 79 nM T89534 C2PGW1 24896626 IC50 = 1440 nM T89534 C06PDG 24952192 Ki = 2300 nM T89534 CG1CF9 24952193 Ki = 5500 nM T89534 CZC7L8 24953162 IC50 > 10000 nM T89534 C4W7BN 24954947 IC50 > 10000 nM T89534 C6XC2R 24954951 IC50 > 20000 nM T89534 CHY0D7 25013322 IC50 > 10000 nM T89534 C0TPS5 25013653 IC50 > 10000 nM T89534 CWU91M 25013811 IC50 > 10000 nM T89534 CSH29L 25013812 IC50 > 10000 nM T89534 C7J6IQ 25027904 EC50 > 100000 nM T89534 C4EGR5 25027907 IC50 = 2950 nM T89534 CDK06N 25027908 IC50 = 1410 nM T89534 CKY0G2 25028122 IC50 = 32100 nM T89534 C2G1JK 25053351 Ki > 30000 nM T89534 CAW8M0 25070694 IC50 > 10000 nM T89534 CYVP87 25110671 IC50 = 8.4 nM T89534 CTYA32 25110672 IC50 = 10.4 nM T89534 CO41GX 25128805 Ki > 1000000 nM T89534 C4EI0A 25128806 Ki > 1000000 nM T89534 CQ34ZE 25128807 IC50 = 2100 nM T89534 CI19MZ 25128808 Ki > 1000000 nM T89534 COWS64 25128809 Ki > 1000000 nM T89534 C42RCW 25128810 Ki > 1000000 nM T89534 C8Q5ZK 25128811 Ki > 1000000 nM T89534 CD3Q4U 25128812 IC50 > 1000000 nM T89534 C6V1ZT 25128813 Ki > 1000000 nM T89534 CAG08U 25128815 IC50 > 1000000 nM T89534 C2FQX9 25128816 IC50 > 1000000 nM T89534 C1HLM6 25129159 Ki > 1000000 nM T89534 C7QFR2 25129160 Ki > 1000000 nM T89534 C1PS3N 25129161 Ki > 1000000 nM T89534 CZS7Q1 25129163 Ki > 1000000 nM T89534 C1XZ5O 25129164 Ki > 1000000 nM T89534 C4YMG0 25129166 Ki > 1000000 nM T89534 CX70KG 25129167 Ki = 2400 nM T89534 CGYS93 25129168 IC50 = 6900 nM T89534 C2E7NK 25129501 Ki > 1000000 nM T89534 CP7YX6 25129502 Ki > 1000000 nM T89534 CTX93Q 25129503 Ki > 1000000 nM T89534 CRA61L 25129504 Ki > 1000000 nM T89534 CV4AP7 25129505 Ki > 1000000 nM T89534 CZF6G7 25129855 Ki > 1000000 nM T89534 CNE47Z 25129856 IC50 = 1800 nM T89534 CC7FL0 25129857 IC50 = 4100 nM T89534 CV0W4X 25129858 IC50 > 1000000 nM T89534 C6W5KP 25129859 IC50 > 1000000 nM T89534 C9Z1YD 25129860 Ki > 1000000 nM T89534 CJ35NZ 25130215 Ki > 1000000 nM T89534 C2X5HD 25130216 Ki > 1000000 nM T89534 C94OVU 25130220 Ki > 1000000 nM T89534 C03ICO 25130561 Ki > 1000000 nM T89534 CZAN43 25130562 IC50 > 1000000 nM T89534 C0IFU7 25130563 IC50 > 1000000 nM T89534 CJT49R 25130564 Ki > 1000000 nM T89534 CRSM67 25130565 IC50 > 1000000 nM T89534 CM8YT4 25130566 IC50 > 1000000 nM T89534 CQ90UO 25130567 Ki > 1000000 nM T89534 COS0E1 25130893 IC50 > 1000000 nM T89534 CR29KD 25130894 IC50 > 1000000 nM T89534 CKX9J5 25130897 Ki > 1000000 nM T89534 CE9LJ6 25130898 Ki > 1000000 nM T89534 CV7WC6 25130899 Ki > 1000000 nM T89534 CJ4AK0 25130900 Ki > 1000000 nM T89534 C7HYX1 25131213 Ki > 1000000 nM T89534 C5PBM7 25131214 Ki = 7200 nM T89534 C14WCP 25131215 IC50 > 1000000 nM T89534 C7MVU3 25131217 Ki > 1000000 nM T89534 C1ZK7W 25131539 IC50 > 1000000 nM T89534 CBGD76 25131540 IC50 = 5500 nM T89534 CX3NA8 25131542 Ki > 1000000 nM T89534 CX12DM 25131544 Ki > 1000000 nM T89534 CIQ2E4 25131893 IC50 = 2100 nM T89534 C28UOB 25131894 IC50 > 1000000 nM T89534 CK2ZT3 25131895 Ki > 1000000 nM T89534 CD13ZC 25131898 IC50 > 1000000 nM T89534 C1UZL6 25132248 Ki > 1000000 nM T89534 CIO06J 25132250 IC50 = 12000 nM T89534 CVFZ60 25132251 Ki > 1000000 nM T89534 CZX45O 25132598 IC50 = 4500 nM T89534 C2ANY3 25132599 Ki > 1000000 nM T89534 CC95RT 25132600 IC50 > 1000000 nM T89534 C27KJG 25132602 IC50 > 1000000 nM T89534 CQNY78 25132933 IC50 = 6900 nM T89534 C6A8WM 25132934 IC50 > 1000000 nM T89534 CO84WJ 25132935 IC50 > 1000000 nM T89534 C6Z4IK 25132936 IC50 > 1000000 nM T89534 C9JI7L 25132937 IC50 > 1000000 nM T89534 CMYZ51 25132938 IC50 > 1000000 nM T89534 CXO4C6 25132939 Ki > 1000000 nM T89534 C9DU6Q 25132940 IC50 > 1000000 nM T89534 CZE3J7 25132941 Ki > 1000000 nM T89534 CR6ME8 25133259 Ki > 1000000 nM T89534 C0ET3J 25133260 Ki > 1000000 nM T89534 CK3VF4 25133261 Ki > 1000000 nM T89534 CB9K2T 25133267 Ki > 1000000 nM T89534 C6ZXQ0 25133268 Ki > 1000000 nM T89534 C9K0ZI 25133269 IC50 > 1000000 nM T89534 C4RG8X 25133607 Ki > 1000000 nM T89534 CD3IH0 25133608 IC50 > 1000000 nM T89534 CI82HF 25133609 IC50 = 9800 nM T89534 CM7VK8 25133611 Ki > 1000000 nM T89534 CD0NT6 25133612 Ki > 1000000 nM T89534 CWC8R0 25133614 IC50 = 5800 nM T89534 C2OCQ5 25133615 Ki = 2400 nM T89534 CEC4P2 25133616 Ki > 1000000 nM T89534 CJ98GU 25133950 Ki > 1000000 nM T89534 C32UKW 25133951 IC50 > 1000000 nM T89534 CE1WN2 25133952 Ki > 1000000 nM T89534 CNU20J 25133953 Ki > 1000000 nM T89534 C0V3KC 25133954 IC50 > 1000000 nM T89534 CLT57Z 25133955 Ki > 1000000 nM T89534 CCW71Z 25133956 Ki > 1000000 nM T89534 CA76HY 25133959 Ki > 1000000 nM T89534 CI3RZ8 25133960 IC50 > 1000000 nM T89534 C21XDY 25145083 Ki > 10000 nM T89534 CLZB04 25147765 IC50 = 37000 nM T89534 C2TJ3P 25191004 IC50 = 1000 nM T89534 C98JQI 25218466 IC50 > 10000 nM T89534 CR8F9X 25218467 IC50 > 10000 nM T89534 C87ARD 25225237 IC50 = 50000 nM T89534 CLY9W3 25235364 IC50 > 10000 nM T89534 C3FW0Y 25257459 IC50 > 10000 nM T89534 CY6X2V 25258136 IC50 = 89 nM T89534 CV4Y6N 25258138 IC50 = 93 nM T89534 CLX0P9 25258381 IC50 > 10000 nM T89534 CNLS64 25258386 IC50 = 3400 nM T89534 CSG7P9 25258611 IC50 = 670 nM T89534 COM4U3 42609838 EC50 = 170000 nM T89534 CH6PI0 43135503 IC50 = 479 nM T89534 CX89HM 44138106 Ki > 5000 nM T89534 C42TWL 44224340 EC50 = 440 nM T89534 C36BKU 44224542 EC50 = 0.11 nM T89534 C0FRP9 44224543 EC50 = 16 nM T89534 CEFT15 44224544 EC50 = 0.11 nM T89534 CLT65I 44225214 EC50 = 10.7 nM T89534 CS5PK0 44225454 EC50 = 20.2 nM T89534 CL1YK5 44225696 EC50 = 2 nM T89534 CFI64J 44227599 EC50 = 330 nM T89534 CXV83I 44227600 EC50 = 65 nM T89534 C40MCV 44275590 IC50 = 366 nM T89534 CY8L2T 44275591 IC50 = 91 nM T89534 CY1O5L 44280253 IC50 = 652 nM T89534 CHWV93 44280284 IC50 = 14 nM T89534 C3DS6O 44280299 IC50 = 490 nM T89534 CB32JI 44280300 IC50 = 89 nM T89534 CP8D0O 44280322 IC50 = 49 nM T89534 CFW6Y4 44280362 IC50 = 531 nM T89534 CTB5L8 44280369 IC50 = 109 nM T89534 C2FE9I 44280602 IC50 = 1415 nM T89534 C5PKE0 44280604 IC50 = 3563 nM T89534 CD94FC 44280669 IC50 = 1050 nM T89534 C7SY2D 44280670 IC50 = 551 nM T89534 C8YM6T 44280672 IC50 = 179 nM T89534 C6UQO3 44280673 IC50 = 68 nM T89534 CFG0A5 44280682 IC50 = 6.7 nM T89534 C9C6HY 44280687 IC50 = 929 nM T89534 C8HK7P 44280689 IC50 = 413 nM T89534 C0LNF3 44280705 IC50 = 71 nM T89534 CEX2O1 44280720 IC50 = 149 nM T89534 CKUI19 44280721 IC50 = 58 nM T89534 CPB4K1 44280724 IC50 = 105 nM T89534 C8QZY6 44283478 EC50 = 770 nM T89534 C9R3AO 44299445 Ki = 37 nM T89534 CT2MK0 44299446 Ki = 170 nM T89534 C5B6IN 44300330 IC50 = 3200 nM T89534 CH4PU5 44305819 IC50 > 10000 nM T89534 CP6A0S 44309223 IC50 = 10 nM T89534 CP52NB 44309415 IC50 = 6.2 nM T89534 CKG5Z0 44317015 IC50 > 5000 nM T89534 C2KD4V 44317238 IC50 = 1260 nM T89534 CPKH32 44317395 IC50 = 1550 nM T89534 C2GZJ0 44317407 IC50 > 5000 nM T89534 CW21CA 44317747 Ki > 10000 nM T89534 C1HK7V 44319061 Ki = 0.36 nM T89534 CE9J8B 44319062 Ki = 2.5 nM T89534 C13KXZ 44319097 Ki = 3.8 nM T89534 CX6S1W 44319117 Ki = 60 nM T89534 C28JXF 44319637 IC50 = 7 nM T89534 C7S5JR 44319707 IC50 = 7.5 nM T89534 C58TKM 44319799 IC50 = 8.8 nM T89534 C7IXG8 44319951 IC50 = 3.9 nM T89534 C8GAE7 44319960 IC50 = 3 nM T89534 C4BID0 44319971 IC50 = 2.6 nM T89534 C4XTK5 44319973 IC50 = 11 nM T89534 CC5QD0 44319981 IC50 = 3 nM T89534 CXZP05 44320014 IC50 = 35 nM T89534 CIC5N6 44320017 IC50 = 542 nM T89534 C7PS6E 44320029 IC50 = 7.4 nM T89534 CMLT05 44320030 IC50 = 490 nM T89534 CRBN05 44325311 IC50 = 5.9 nM T89534 CD0IH3 44325322 IC50 = 112 nM T89534 CNP05V 44325337 IC50 = 2 nM T89534 COTS43 44325352 IC50 = 120 nM T89534 C2B1OU 44325368 IC50 = 20.1 nM T89534 CZ9Y1O 44325433 IC50 > 3200 nM T89534 C5V7WZ 44325464 IC50 = 8 nM T89534 CS3R4P 44325467 IC50 = 53.1 nM T89534 C6NAY0 44325476 IC50 = 44.3 nM T89534 COL02R 44325510 IC50 = 341.9 nM T89534 CZ0P9W 44325539 IC50 = 34.9 nM T89534 CR94YN 44325546 IC50 = 25 nM T89534 C6TZA9 44325547 IC50 = 0.51 nM T89534 CML6J0 44325551 IC50 = 1.2 nM T89534 CL95JC 44325552 IC50 = 4.7 nM T89534 CDK3S0 44325556 IC50 = 0.5 nM T89534 CH8P0Z 44325557 IC50 = 23.1 nM T89534 C9DA8B 44325570 IC50 = 1 nM T89534 C6B7RO 44325581 IC50 = 0.8 nM T89534 C49BSH 44325582 IC50 = 14.8 nM T89534 CDX49O 44325585 IC50 = 13.5 nM T89534 CEAL30 44325586 IC50 = 5.3 nM T89534 CISM83 44325587 IC50 = 5.3 nM T89534 C8LG6M 44325589 IC50 = 1.3 nM T89534 C4K0RZ 44325613 IC50 = 1.4 nM T89534 CVD76C 44325614 IC50 = 41.1 nM T89534 CXYC85 44325632 IC50 = 3.4 nM T89534 CAE3Y9 44325639 IC50 = 0.8 nM T89534 C4S9ZI 44325650 IC50 = 1.2 nM T89534 CMJ0Z5 44325659 IC50 = 4.7 nM T89534 CEN5R9 44325692 IC50 = 1 nM T89534 CD9P3O 44343122 EC50 = 4 nM T89534 CQ7V0U 44343261 EC50 > 10000 nM T89534 C1SG7C 44348079 IC50 = 0.7 nM T89534 CSVW34 44348099 IC50 = 4.4 nM T89534 C1H7MO 44348132 IC50 = 1 nM T89534 CE4YL7 44348273 IC50 = 4 nM T89534 C28EVO 44348377 IC50 = 155 nM T89534 C2GL8B 44348457 IC50 = 21 nM T89534 CXY05L 44348479 IC50 = 3.6 nM T89534 CWCS52 44348487 IC50 = 4 nM T89534 CQA68R 44348495 IC50 = 3.6 nM T89534 CE3O6Y 44348510 IC50 = 15 nM T89534 C0I9FH 44348522 IC50 = 1.4 nM T89534 CLX35U 44348531 IC50 = 1.7 nM T89534 CX82TV 44348539 IC50 = 1 nM T89534 C90INV 44348540 IC50 = 2.3 nM T89534 C3B6LK 44355916 EC50 = 0.064 nM T89534 CK1UW9 44355917 EC50 = 5.2 nM T89534 CBO3X2 44355927 EC50 = 130 nM T89534 CIWX06 44356135 EC50 = 150 nM T89534 CW67AN 44356136 EC50 = 14 nM T89534 CM7H1I 44356536 EC50 = 73 nM T89534 C7UH6W 44356621 Ki = 13 nM T89534 CYBO90 44356823 Ki = 24 nM T89534 C4UTM7 44356833 Ki = 23 nM T89534 CT07FI 44389476 EC50 = 141 nM T89534 CG80UZ 44389487 EC50 = 21 nM T89534 CL92HF 44389493 EC50 = 59 nM T89534 COW1E9 44389558 EC50 = 19 nM T89534 C5ECY2 44389569 EC50 = 92 nM T89534 CY5K2O 44389570 EC50 = 173 nM T89534 CRN5I1 44389572 EC50 = 143 nM T89534 CL7C9P 44389577 EC50 = 2411 nM T89534 CZJ5C4 44389581 EC50 = 1.6 nM T89534 C9Q4UB 44389582 EC50 = 1 nM T89534 CSP4T9 44389593 EC50 = 137 nM T89534 CEHT06 44389595 EC50 = 0.6 nM T89534 CTJ9Q6 44389606 EC50 = 743 nM T89534 CS47PF 44389609 EC50 = 2.6 nM T89534 CUA5F4 44389617 EC50 = 36 nM T89534 CVT09Q 44389633 EC50 = 336 nM T89534 CV24GJ 44389648 EC50 = 1980 nM T89534 C8MI1L 44389650 EC50 = 203 nM T89534 C9RUX6 44389654 EC50 = 43 nM T89534 CL2W9P 44389655 EC50 = 68 nM T89534 CQ01VW 44389659 EC50 = 50 nM T89534 C2PDC8 44389876 IC50 = 0.86 nM T89534 C8ZIP3 44389878 IC50 = 1.72 nM T89534 CA05VL 44389880 IC50 = 2.12 nM T89534 CB1H3E 44389883 IC50 = 1.39 nM T89534 CUP57N 44389890 IC50 = 14.46 nM T89534 CBIA52 44389891 IC50 = 2.15 nM T89534 CQU8C6 44389896 IC50 = 2.65 nM T89534 C10LSB 44389901 IC50 = 3.05 nM T89534 C6CIB9 44389904 IC50 = 1.43 nM T89534 C8YNX2 44389906 IC50 = 0.22 nM T89534 C39DPH 44389907 IC50 = 3.58 nM T89534 C2ZS9G 44389914 IC50 = 2.74 nM T89534 C19MKQ 44389919 IC50 = 3.94 nM T89534 C4W5VU 44389922 IC50 = 0.43 nM T89534 CB7K5Y 44389934 IC50 = 0.46 nM T89534 CVG41F 44389943 IC50 = 0.27 nM T89534 CO1H5G 44389945 IC50 = 1.08 nM T89534 C8GD3V 44389948 IC50 = 0.22 nM T89534 CP0Y8G 44390069 IC50 = 1.4 nM T89534 C1JQD2 44390070 IC50 = 38 nM T89534 CPFB84 44390071 IC50 = 0.3 nM T89534 C24ZDP 44390072 IC50 = 0.9 nM T89534 CXHL23 44390084 IC50 = 14 nM T89534 CQ92BW 44390097 IC50 = 0.9 nM T89534 C6RC2Y 44390116 IC50 = 45 nM T89534 C4GP0U 44390120 IC50 = 0.8 nM T89534 C1DS5R 44390163 IC50 = 0.8 nM T89534 C7ZQ1J 44391057 IC50 = 39 nM T89534 C50XAP 44391076 IC50 = 13 nM T89534 C5Y6CT 44391206 IC50 = 2.4 nM T89534 C0ZIT7 44391782 IC50 = 0.3 nM T89534 CS4XD9 44391788 IC50 = 6.3 nM T89534 CV4G0H 44391842 IC50 = 0.7 nM T89534 CRJE53 44391854 IC50 = 0.4 nM T89534 C5W2IH 44391860 IC50 = 2.5 nM T89534 CZOJ29 44391870 IC50 = 0.5 nM T89534 CIT5P8 44391879 IC50 = 1.7 nM T89534 C0B5IT 44391881 IC50 = 0.7 nM T89534 CZH85I 44391888 IC50 = 1.2 nM T89534 CQD42M 44391889 IC50 = 0.9 nM T89534 CT0BO6 44391890 IC50 = 0.8 nM T89534 C1NIS3 44391905 IC50 = 0.7 nM T89534 C74EHI 44391917 IC50 = 0.5 nM T89534 CP15SF 44392410 IC50 = 19.82 nM T89534 CA82NU 44392580 IC50 = 990 nM T89534 CC72ZY 44392593 IC50 = 335 nM T89534 CDMN93 44392636 IC50 = 12 nM T89534 CS8ZN5 44393200 IC50 = 1.2 nM T89534 CP53NK 44393219 IC50 = 0.8 nM T89534 CB5DS4 44393237 IC50 = 1 nM T89534 C1GA9N 44393240 IC50 = 1.7 nM T89534 C0TLH5 44393249 IC50 = 2.2 nM T89534 CL27NW 44393263 IC50 = 0.3 nM T89534 CR64AD 44393267 IC50 = 0.5 nM T89534 CTN81R 44393286 IC50 = 0.9 nM T89534 CW59RL 44393287 IC50 = 2.5 nM T89534 C01ODV 44393310 IC50 = 0.6 nM T89534 C82WUF 44393322 IC50 = 2 nM T89534 CO1Q0W 44393335 IC50 = 0.6 nM T89534 C0JXU4 44393336 IC50 = 1.5 nM T89534 CC89WN 44393340 IC50 = 0.4 nM T89534 C2WXI0 44393342 IC50 = 3.9 nM T89534 CNP73S 44393366 IC50 = 0.6 nM T89534 C8E0AJ 44393367 IC50 = 2.2 nM T89534 CQY82B 44393380 IC50 = 0.6 nM T89534 CP25CW 44393381 IC50 = 1.8 nM T89534 C8P3FU 44393399 IC50 = 1.3 nM T89534 CIS79C 44393400 IC50 = 2 nM T89534 C1XOK4 44393405 IC50 = 0.5 nM T89534 CV5YB6 44393408 IC50 = 7.3 nM T89534 CRB41V 44393419 IC50 = 16 nM T89534 C5U2KP 44394160 IC50 = 209 nM T89534 C13SYV 44396250 Ki = 19 nM T89534 CB1P0S 44396251 Ki = 8.8 nM T89534 CHY1C3 44396271 Ki = 72 nM T89534 C29MBI 44396272 Ki = 11 nM T89534 C4TQ6N 44396282 Ki = 11 nM T89534 CH2Y3L 44396283 Ki = 6.2 nM T89534 CWZB52 44396284 Ki = 140 nM T89534 CD80LM 44396296 Ki = 34 nM T89534 C6SI5L 44396297 Ki > 200 nM T89534 C45LRH 44396317 Ki = 10 nM T89534 C5JG6H 44396330 Ki = 46 nM T89534 CA8V4G 44396331 Ki = 94 nM T89534 CD2EY3 44399091 IC50 > 5000 nM T89534 CDJ7H0 44399199 IC50 = 1800 nM T89534 CK1X0O 44400690 IC50 = 877 nM T89534 CSE07P 44402388 IC50 = 3.34 nM T89534 CSZ2J0 44402418 IC50 = 31.2 nM T89534 C6I3PD 44402432 IC50 = 27.2 nM T89534 C3FR5B 44402483 IC50 = 18 nM T89534 C6CWQ3 44402516 IC50 = 10 nM T89534 CC3QK6 44402532 IC50 = 57.4 nM T89534 CM35QL 44402545 IC50 = 18 nM T89534 CL9CQ8 44402598 IC50 = 51.4 nM T89534 CN57AQ 44402634 IC50 = 126 nM T89534 CQH5B1 44402654 IC50 = 6 nM T89534 CF0VN8 44402705 IC50 = 39 nM T89534 C7VCZ5 44402711 IC50 > 10000 nM T89534 CXI97U 44402746 IC50 > 10000 nM T89534 CGRX27 44402769 IC50 > 10000 nM T89534 C9XS4E 44402799 IC50 > 10000 nM T89534 CB2V0A 44403942 Ki = 7.3 nM T89534 CARV69 44405133 IC50 = 0.6 nM T89534 CKZ15D 44405150 IC50 = 0.5 nM T89534 CR4V3M 44405163 IC50 = 0.6 nM T89534 C2C9OW 44405166 IC50 = 0.2 nM T89534 CG85OU 44405167 IC50 = 0.5 nM T89534 CLE8X1 44405174 IC50 = 0.4 nM T89534 C72SFE 44405903 IC50 = 1730 nM T89534 CB56DO 44407581 IC50 = 830 nM T89534 CWT4M0 44407582 EC50 = 830 nM T89534 C1ISP9 44407583 EC50 = 153 nM T89534 C5WQ6O 44407584 IC50 = 16 nM T89534 CP5DT4 44407585 IC50 = 14 nM T89534 C2A5EY 44407586 EC50 = 12 nM T89534 C79JEI 44407631 EC50 = 160 nM T89534 CB0L6S 44407636 EC50 = 1000 nM T89534 C2W0PF 44407655 EC50 > 1000 nM T89534 CA7S2Z 44407657 EC50 = 378 nM T89534 CWU1O4 44407658 IC50 = 5155 nM T89534 CP7CQ0 44407661 EC50 = 480 nM T89534 CNC2A4 44407662 IC50 = 26 nM T89534 CCPB47 44407663 IC50 = 60 nM T89534 C8Y7ZB 44407724 IC50 = 328 nM T89534 C5QW0O 44407725 EC50 = 1391 nM T89534 C3LGU8 44407741 IC50 = 892 nM T89534 C6J3VA 44407760 EC50 = 3237 nM T89534 C1O6WJ 44407763 EC50 = 583 nM T89534 C21CBM 44407771 EC50 = 844 nM T89534 CD3E0R 44407782 EC50 > 1000 nM T89534 C2O1DA 44407785 IC50 = 3984 nM T89534 C2POZ8 44407805 IC50 = 109 nM T89534 CQ1Y0R 44407807 EC50 = 161 nM T89534 CZ0XT5 44407808 EC50 = 144 nM T89534 CF5Z0G 44407811 EC50 = 650 nM T89534 CF0AQ2 44407812 EC50 = 243 nM T89534 CN06HP 44407826 IC50 = 253 nM T89534 CUA05F 44407827 EC50 = 63 nM T89534 CXD31Y 44407857 EC50 > 1000 nM T89534 C4K3ZG 44408764 IC50 = 157 nM T89534 C7CSE3 44408771 IC50 = 5460 nM T89534 CF06GJ 44408808 IC50 = 524 nM T89534 C1K3FC 44409005 IC50 = 229 nM T89534 C5HM2W 44409078 IC50 = 1090 nM T89534 CIUR71 44409233 IC50 > 10000 nM T89534 CF0IQ7 44412807 IC50 > 10000 nM T89534 CI4KN9 44412821 IC50 = 1420 nM T89534 C5E9XO 44412823 IC50 = 880 nM T89534 C5S9OV 44412835 IC50 = 3740 nM T89534 CN9X6E 44412848 IC50 > 10000 nM T89534 CE60QX 44412849 IC50 = 481 nM T89534 CZ13IC 44412903 IC50 = 113 nM T89534 C3ADY8 44412904 IC50 = 389 nM T89534 CJ4S8E 44412954 IC50 = 4245 nM T89534 C0JAX2 44412955 IC50 > 10000 nM T89534 C4EZB6 44412956 IC50 = 319 nM T89534 CW08IO 44412979 IC50 = 6450 nM T89534 CFH31O 44412983 IC50 = 79 nM T89534 C5RT0I 44413033 IC50 = 567 nM T89534 C2TFX6 44413049 IC50 > 10000 nM T89534 CE2P7W 44413050 IC50 = 4023 nM T89534 CQW1N9 44414035 IC50 = 46 nM T89534 CXBZ80 44414036 EC50 = 33.1 nM T89534 C2H8RD 44414046 IC50 = 93 nM T89534 CQC9F4 44414050 EC50 = 1170 nM T89534 CIS2L0 44414060 EC50 = 152 nM T89534 CJBQ27 44414066 EC50 = 61 nM T89534 C09CRE 44414068 IC50 = 1478 nM T89534 CECT78 44414069 IC50 = 2080 nM T89534 CI12OU 44414094 EC50 = 50 nM T89534 CF5T6Y 44414110 IC50 = 176 nM T89534 CGP27O 44414111 IC50 = 470 nM T89534 CXG13L 44414126 EC50 = 104 nM T89534 C8E5PN 44414131 EC50 = 65 nM T89534 CV1LR4 44414182 IC50 = 230 nM T89534 CALJ60 44414245 IC50 = 23 nM T89534 C5WTR2 44414246 IC50 = 49.2 nM T89534 C7MT9J 44414260 IC50 = 139 nM T89534 CL0K4C 44414274 IC50 = 40 nM T89534 C90LXU 44414284 EC50 = 1100 nM T89534 C0I3YZ 44414292 IC50 = 422 nM T89534 CPFS03 44414293 IC50 = 82 nM T89534 C7L2PW 44415352 IC50 = 1210 nM T89534 C2Y9BF 44415353 IC50 = 455 nM T89534 C96JSR 44415397 IC50 = 3900 nM T89534 C5V2SP 44415478 IC50 = 97 nM T89534 C7YQ9X 44415498 IC50 = 414 nM T89534 CREK89 44415499 IC50 = 146 nM T89534 C18JCA 44415511 IC50 = 310 nM T89534 CGS79I 44415523 IC50 = 84 nM T89534 C1FCL0 44415547 IC50 = 605 nM T89534 C6PD3R 44415553 EC50 = 169 nM T89534 CH50DC 44415571 EC50 = 79 nM T89534 CSF5O8 44415669 EC50 = 241 nM T89534 C7C4XF 44415699 EC50 = 391 nM T89534 CCO34X 44415700 EC50 = 30 nM T89534 C3KI0H 44415761 IC50 > 10000 nM T89534 CV37CW 44415788 EC50 = 140 nM T89534 C9T3QO 44423844 EC50 = 100 nM T89534 CG72WC 44427370 Ki = 0.4 nM T89534 C2F8CW 44427371 Ki = 0.73 nM T89534 CHB94D 44427372 Ki = 0.24 nM T89534 CYB7J6 44427373 Ki = 0.18 nM T89534 CQ96LY 44427374 Ki = 0.2 nM T89534 CN2M3P 44427375 Ki = 1.09 nM T89534 CQ74SE 44427404 Ki = 0.091 nM T89534 CHK6A4 44427405 Ki = 0.48 nM T89534 CL1Y4N 44430357 IC50 = 3300 nM T89534 C5S6XP 44430360 IC50 = 2470 nM T89534 CUQT28 44430361 IC50 > 5000 nM T89534 CKF6I1 44430362 IC50 > 5000 nM T89534 COT67E 44430364 IC50 = 802 nM T89534 C2YF4G 44430366 IC50 = 2640 nM T89534 CBGX08 44430369 IC50 > 5000 nM T89534 CY4XR5 44430372 IC50 = 21 nM T89534 C27KUN 44430374 IC50 = 802 nM T89534 C6LV9A 44430376 IC50 = 53 nM T89534 CHM5G2 44430378 IC50 > 5000 nM T89534 C4ERT8 44433138 Ki = 7100 nM T89534 C9EK6V 44433139 Ki = 12000 nM T89534 CEJ8B1 44433140 Ki = 32000 nM T89534 CNX1A6 44433141 Ki = 7900 nM T89534 C2J1PU 44433142 Ki = 38000 nM T89534 C3SJ5V 44433504 Ki > 1100 nM T89534 CJ5G2Z 44439806 IC50 = 11 nM T89534 CG17VZ 44439807 IC50 = 1 nM T89534 C5Y4CM 44439809 IC50 = 37 nM T89534 C28PCX 44439811 IC50 = 1134 nM T89534 C4WS3E 44439813 IC50 = 378 nM T89534 C3H6BA 44439815 IC50 = 40 nM T89534 C3DGB7 44439820 IC50 = 31 nM T89534 CL9IE2 44439822 IC50 = 6.6 nM T89534 C7RLX5 44439823 IC50 = 13 nM T89534 C1A0PH 44439825 IC50 = 10.1 nM T89534 C3KS9O 44439826 IC50 = 22 nM T89534 CFZ0N1 44439827 IC50 = 9.1 nM T89534 CMW5Z8 44439828 IC50 = 440 nM T89534 CWBD12 44439829 IC50 = 69 nM T89534 C2Y4GR 44439830 IC50 = 23 nM T89534 CZNS72 44439831 IC50 = 13 nM T89534 COGW71 44439832 IC50 = 20 nM T89534 C76TMP 44439833 IC50 = 175 nM T89534 C82NQD 44439834 IC50 = 7.8 nM T89534 C98BPO 44439835 IC50 = 4.9 nM T89534 C1HZ2K 44439836 IC50 = 4 nM T89534 C3LO1U 44440237 EC50 = 980 nM T89534 CLK05T 44440238 IC50 = 2330 nM T89534 CP3JU8 44440239 EC50 > 1000 nM T89534 C34ERB 44440240 EC50 = 4893 nM T89534 C5KG7L 44440241 EC50 = 1300 nM T89534 CB1ZS3 44440262 EC50 = 44 nM T89534 CKON02 44440263 EC50 = 435 nM T89534 C5DB8N 44440264 EC50 > 1000 nM T89534 C89JEW 44440265 EC50 > 1000 nM T89534 CR7G2K 44440266 EC50 > 1000 nM T89534 CVT4O9 44440267 EC50 > 1000 nM T89534 CO98DZ 44440268 EC50 > 1000 nM T89534 CC73BF 44440269 EC50 = 407 nM T89534 C6O5DS 44441690 Ki = 37 nM T89534 C8YOH7 44441691 Ki = 100 nM T89534 CG6W1K 44441692 Ki = 35 nM T89534 C5OMR2 44441693 Ki = 75 nM T89534 CKQ1H7 44441694 Ki = 332 nM T89534 CEMX26 44441695 Ki = 63052 nM T89534 C5WVG8 44441696 Ki = 382 nM T89534 CY32PU 44441697 Ki = 17879 nM T89534 CL3WI5 44441857 IC50 = 5300 nM T89534 CIL2C9 44441858 EC50 > 1000 nM T89534 CR2S3A 44441859 IC50 = 3110 nM T89534 C6GRK9 44441860 EC50 > 1000 nM T89534 C2FC5N 44441861 EC50 = 820 nM T89534 CA1BY2 44441862 IC50 = 4380 nM T89534 C6SMB2 44441863 EC50 = 490 nM T89534 CTQ15A 44441864 EC50 > 1000 nM T89534 CF06VH 44441865 EC50 = 130 nM T89534 C1X5MS 44441866 EC50 = 430 nM T89534 CYG7X4 44473146 IC50 > 10000 nM T89534 CT0B2Q 44473422 EC50 > 1000 nM T89534 CR5SI0 44476535 EC50 > 10000 nM T89534 CM29JD 44516036 IC50 > 10000 nM T89534 C3ND5A 44542643 EC50 > 1000 nM T89534 C3SBL5 44543099 EC50 > 1000 nM T89534 CK8MH3 44565647 Ki = 26300 nM T89534 CEI26D 44569027 Ki > 1000000 nM T89534 CCPW27 44569028 IC50 > 1000000 nM T89534 CF4RS6 44569029 Ki = 7500 nM T89534 CEA0U9 44579680 Ki = 55 nM T89534 C8W6ZF 44580025 Ki = 977 nM T89534 CXGP15 44580026 Ki = 724 nM T89534 CW5O3K 44580027 Ki = 158 nM T89534 C2L3NV 44588414 IC50 = 16000 nM T89534 C3TRJ2 44589610 EC50 = 10 nM T89534 CZOU20 44589952 IC50 = 8.77 nM T89534 CNM79D 44589953 IC50 = 1.9 nM T89534 C1JCM3 44589998 IC50 = 6.7 nM T89534 CDP6W8 44589999 IC50 = 10.3 nM T89534 C5FC9V 44590000 IC50 = 16.2 nM T89534 CYI29S 44590098 IC50 = 14 nM T89534 CD8R7Y 44590099 IC50 = 126 nM T89534 C7T8KP 44590100 IC50 > 15000 nM T89534 C4RZX5 44590136 IC50 = 6.5 nM T89534 C6NZW2 44590137 IC50 = 5.57 nM T89534 CL7IT6 44592556 IC50 > 100000 nM T89534 CJ3VI8 44593465 Ki > 5000 nM T89534 C6NXD9 44593529 IC50 = 5500 nM T89534 CKYW84 44596355 IC50 = 1200 nM T89534 CY0U6X 44596356 IC50 = 150 nM T89534 CQG0F7 44596357 IC50 > 1000 nM T89534 CSR28W 44596358 IC50 > 1000 nM T89534 CAG36H 44596359 IC50 = 16 nM T89534 C6AZU3 44596467 IC50 = 5 nM T89534 C49XRU 44596468 IC50 = 293 nM T89534 C1YRA4 44596469 IC50 = 1210 nM T89534 CS12MF 44596470 IC50 = 1570 nM T89534 C2K1DR 44596471 IC50 = 3.3 nM T89534 C3LMA0 44596573 IC50 = 180 nM T89534 C3KH5Y 44596574 IC50 = 85 nM T89534 CJM37H 44596575 IC50 = 100 nM T89534 C8GJ9B 44596686 IC50 = 3.4 nM T89534 CSQ10X 44596687 IC50 = 190 nM T89534 CFJE97 44596688 IC50 = 13 nM T89534 CYX0C2 44596789 IC50 = 11.1 nM T89534 CM67OY 44596790 IC50 = 4.2 nM T89534 CUT7N3 44596791 IC50 = 6.3 nM T89534 CAI8D6 44596792 IC50 > 10000 nM T89534 C9KW4Y 44596793 IC50 = 687 nM T89534 CBLN03 44596894 IC50 > 1000 nM T89534 CX76YZ 44596895 IC50 = 9 nM T89534 CLWY41 44596896 IC50 = 4 nM T89534 CSUT20 44596897 IC50 = 35 nM T89534 CRUO49 44596898 IC50 > 1000 nM T89534 C1FI6O 44596992 IC50 = 4.5 nM T89534 C0YUC1 44596993 IC50 = 6.3 nM T89534 CN1M3J 44596994 IC50 = 128 nM T89534 C6NEV4 44596995 IC50 = 150 nM T89534 C42NEY 44596996 IC50 = 2.5 nM T89534 CUK16W 44597094 IC50 = 122 nM T89534 C43LCQ 44597095 IC50 = 10 nM T89534 CLJM84 44597096 IC50 = 161 nM T89534 C9R2CP 44597097 IC50 = 111 nM T89534 CL01OK 44597098 IC50 = 312 nM T89534 CMR68J 44597209 IC50 = 6.2 nM T89534 CWG9Z7 44597210 IC50 = 40.97 nM T89534 CYA0B6 44597211 IC50 = 580 nM T89534 CE31LY 44597212 IC50 = 590 nM T89534 C9QO1F 44597743 IC50 = 293 nM T89534 C63LWP 44597744 IC50 = 5.4 nM T89534 C3O2NE 44597745 IC50 = 217 nM T89534 CME14J 44597857 IC50 = 1.2 nM T89534 CI9E7J 44597858 IC50 = 1.6 nM T89534 C95YGF 44597859 IC50 = 1.2 nM T89534 CD9EL6 44597860 IC50 = 8.7 nM T89534 C6GWQ8 44597861 IC50 = 4.8 nM T89534 CS79YT 44597968 IC50 = 2.63 nM T89534 CUO92A 44597969 IC50 = 310 nM T89534 CMXI54 44597970 IC50 = 326 nM T89534 CT9Q0J 44597971 IC50 = 4.8 nM T89534 CSOD50 44597973 IC50 = 120 nM T89534 CIJP09 44605898 EC50 > 10000 nM T89534 C9PLK4 45263610 IC50 > 2000 nM T89534 C78JKD 45265930 IC50 > 2000 nM T89534 CN4IE3 45275362 IC50 = 8.1 nM T89534 C4A2MR 46190224 IC50 = 24400 nM T89534 CKX73S 46190225 IC50 = 7600 nM T89534 CJ3Z5R 46231169 EC50 = 27 nM T89534 C9CL7N 46231170 EC50 = 300 nM T89534 C3O2GA 46231223 EC50 = 4000 nM T89534 CR6XM0 46231224 EC50 = 2 nM T89534 C51IGU 46231225 EC50 = 4000 nM T89534 C0ZBS6 46231226 EC50 = 27 nM T89534 C4M9KI 46231227 EC50 = 1500 nM T89534 CJ84WL 46231228 EC50 = 2600 nM T89534 C5C8ZD 46237712 EC50 = 14.06 nM T89534 CP1VU0 46237713 IC50 = 243.22 nM T89534 C0HMU5 46237838 EC50 = 16.48 nM T89534 C6RZX9 46237839 EC50 = 6.918 nM T89534 CKBD82 46237840 EC50 = 92.04 nM T89534 CPD64X 46237841 EC50 = 35.97 nM T89534 C2S6PL 46834818 IC50 > 10000 nM T89534 CL6SY4 46866497 IC50 > 30000 nM T89534 CO1T3Q 46871902 IC50 = 57200 nM T89534 C9UZ5N 46871916 IC50 = 151100 nM T89534 CAYW93 46880832 Ki = 29000 nM T89534 CDHA57 46880834 IC50 > 30000 nM T89534 C72MUY 46889765 IC50 > 5000 nM T89534 C6DVO1 46889848 IC50 > 10000 nM T89534 CZ90FC 46894119 IC50 > 25000 nM T89534 C3Q7RI 46913890 IC50 > 4960 nM T89534 CX70GY 46915355 IC50 > 10000 nM T89534 CN9L7G 46916268 IC50 = 2200 nM T89534 C0FNE4 46916592 IC50 = 3.7 nM T89534 CYVP45 46916643 IC50 = 3.8 nM T89534 C05YMH 46935020 IC50 = 82 nM T89534 CL7P3N 46938234 IC50 > 10000 nM T89534 CX0NO8 49782554 EC50 < 15848.93 nM T89534 CC7T8Q 49782555 EC50 = 1655.77 nM T89534 CD07EV 49782777 EC50 < 15848.93 nM T89534 C43UKW 49782778 IC50 < 15848.93 nM T89534 C2JTF0 49782779 EC50 = 1028.02 nM T89534 CS7KX9 49782780 IC50 < 15848.93 nM T89534 C36RYU 49782781 EC50 = 402.72 nM T89534 C8OA0C 49782985 IC50 < 15848.93 nM T89534 C5Y6QU 49782986 EC50 = 35.48 nM T89534 CB8V7R 49782987 EC50 = 9954.05 nM T89534 CU3S6H 49836028 Ki > 50000 nM T89534 C96SLW 49851364 Ki > 100000 nM T89534 CDN4K6 49851369 Ki > 50000 nM T89534 C4YXN1 49851467 Ki > 50000 nM T89534 CUD91T 49862248 EC50 = 1043000 nM T89534 C0SY6G 49864608 EC50 = 0.24 nM T89534 C2JAP4 50919273 EC50 = 20000 nM T89534 C0BPT6 50919274 EC50 = 1870 nM T89534 CY10IC 50940834 EC50 > 10000 nM T89534 CTH45Q 52918523 IC50 > 10000 nM T89534 CF16DR 52937206 EC50 = 340000 nM T89534 CG7LY6 52937207 EC50 = 2300 nM T89534 CS0UY6 52937307 EC50 = 6200 nM T89534 CB94DP 52937308 EC50 = 700000 nM T89534 C75SPY 52937309 EC50 = 600000 nM T89534 CFNK21 52946352 IC50 = 310 nM T89534 CF4W1S 53262779 IC50 = 1000000 nM T89534 CA3SG5 53262780 IC50 = 80000 nM T89534 C83ZHQ 53262781 IC50 = 2800000 nM T89534 C8MU3A 53322265 IC50 > 10000 nM T89534 CYA61L 53323081 EC50 = 7 nM T89534 CEW0A8 53324900 IC50 = 8360 nM T89534 CJCP75 53359074 Ki > 75000 nM T89534 CZQ09C 53465819 IC50 = 1100 nM T89534 CWHK62 53483961 EC50 > 5400 nM T89534 C87KXG 54584962 IC50 = 3500000 nM T89534 C30XLO 54592009 IC50 > 10000 nM T89534 C5ZX4B 54597874 IC50 > 10000 nM T89534 C6ST8W 54675748 IC50 = 0.2 nM T89534 CDI89A 54765689 IC50 = 0.2 nM T89534 CB8U5G 54765691 IC50 = 0.3 nM T89534 CX0Q9I 54765856 IC50 = 0.2 nM T89534 C8O3BH 54765858 IC50 = 0.2 nM T89534 CPM43H 54765860 IC50 = 0.2 nM T89534 C4XG5H 54766021 IC50 = 0.2 nM T89534 CRLE21 54766022 IC50 = 0.2 nM T89534 C7CBA8 54766023 IC50 = 0.2 nM T89534 CJ2K9E 54766174 IC50 = 0.2 nM T89534 C3CNJ8 54766175 IC50 = 0.4 nM T89534 CLP3H4 54766176 IC50 = 0.3 nM T89534 CY5QJ4 54766177 IC50 = 0.1 nM T89534 CR5T9O 54766178 IC50 = 9.7 nM T89534 C90PVJ 54766328 IC50 = 0.4 nM T89534 CL38TD 54766331 IC50 = 0.4 nM T89534 CPH2W0 54766478 IC50 = 0.4 nM T89534 CRP5Z2 54766481 IC50 = 0.4 nM T89534 CHG78U 54766482 IC50 = 0.2 nM T89534 C8AUT4 54766633 IC50 = 0.3 nM T89534 CT7D3W 54766636 IC50 = 0.9 nM T89534 CMO2X4 54766789 IC50 = 0.5 nM T89534 CNUM98 54766945 IC50 = 0.1 nM T89534 C8GR2U 54767099 IC50 = 0.3 nM T89534 C3X1IA 54767260 IC50 = 5.7 nM T89534 C9W5DZ 56593984 Ki > 75000 nM T89534 C8GP2M 56658858 EC50 > 2680 nM T89534 C0HMP7 56662184 EC50 = 357 nM T89534 CH65JX 56662340 EC50 = 2310 nM T89534 C1WS4G 56662341 EC50 > 6510 nM T89534 CWY30K 56665645 EC50 = 3500 nM T89534 C1O0XA 56666151 IC50 = 1.11 nM T89534 CFQ51I 56672695 EC50 = 3800 nM T89534 C9CXS4 56675930 EC50 > 3200 nM T89534 CZT8H6 56676055 EC50 > 1100 nM T89534 C9ZJ8I 56679386 EC50 > 4560 nM T89534 CP06XK 56679387 EC50 > 10000 nM T89534 CP58AC 56679388 EC50 > 10000 nM T89534 CK1N6F 56682681 EC50 > 2610 nM T89534 CG8J9I 56682682 EC50 > 4800 nM T89534 C67XZQ 56927060 EC50 = 2.6 nM T89534 C51ZSU 56940798 EC50 = 0.7 nM T89534 CGK89W 56940799 EC50 = 2 nM T89534 CURV45 56940800 EC50 = 14 nM T89534 C3F0IO 56940801 EC50 = 0.8 nM T89534 C80ZVD 56940946 EC50 = 4 nM T89534 CR4TO6 56941387 EC50 = 3 nM T89534 CZ3DB1 56941388 EC50 = 49 nM T89534 C48FPW 56941825 EC50 = 4 nM T89534 CUQ8X4 56941959 EC50 = 11 nM T89534 CZD36T 56941964 EC50 = 15 nM T89534 C5UK3N 56942100 EC50 = 6 nM T89534 CUB7H1 56942101 EC50 = 28 nM T89534 CGY2K5 56942102 EC50 = 36 nM T89534 COA86V 56942249 EC50 = 3 nM T89534 CBX8N7 56942543 EC50 = 957 nM T89534 CK1G7N 56943018 EC50 = 10 nM T89534 C53OZE 56945585 EC50 = 6.2 nM T89534 C37IJX 57392620 Ki = 1 nM T89534 CF83VM 57401459 Ki > 75000 nM T89534 CTM6K5 57690900 IC50 > 5000 nM T89534 C87TXE 57992044 EC50 > 10000 nM T89534 CI6XF5 58742295 IC50 > 3200 nM T89534 CYI71B 58902727 EC50 > 10000 nM T89534 CE18JH 60202715 EC50 = 27 nM T89534 CE0SK2 66574394 IC50 < 100000 nM T89534 C26BLT 66792935 EC50 = 0.9 nM T89534 CK7C3F 66793234 EC50 = 1 nM T89534 C7D5KR 66793358 EC50 = 27 nM T89534 CW5I4N 66800025 EC50 = 200 nM T89534 CS2XF1 66800044 EC50 = 5.9 nM T89534 CC4D3G 66800191 EC50 = 22 nM T89534 CU3CO9 66800285 EC50 = 357 nM T89534 C8FG7K 66800295 EC50 = 23 nM T89534 CXA2F8 66800317 EC50 = 57 nM T89534 CVH2W8 66800328 EC50 = 6 nM T89534 C2LN5Q 66800382 EC50 = 240 nM T89534 CV63IY 66800384 EC50 = 460 nM T89534 CZLD42 66800405 EC50 = 150 nM T89534 CIGK37 66800456 EC50 = 0.7 nM T89534 CANS48 66801915 EC50 = 350 nM T89534 CRE4B8 66802205 EC50 = 6280 nM T89534 C3Z7JY 66802304 EC50 = 260 nM T89534 C3SKM2 66802363 EC50 = 110 nM T89534 CPU8J0 66802555 EC50 = 1130 nM T89534 C8C4HE 66802616 EC50 = 110 nM T89534 CZ69XC 66802706 EC50 = 101 nM T89534 C6ZF2N 66802727 EC50 = 340 nM T89534 CN07XA 66802737 EC50 > 500 nM T89534 CF3G2U 66802742 EC50 = 1.5 nM T89534 CI1G8L 66802787 EC50 > 500 nM T89534 CZ8KP0 66802802 EC50 = 160 nM T89534 CF1WN2 66803137 EC50 = 2 nM T89534 C24JEX 66803231 EC50 = 8 nM T89534 CBO20T 66803277 EC50 = 0.5 nM T89534 C2F5TS 68037237 EC50 = 17 nM T89534 CMT2I3 68321354 IC50 = 280 nM T89534 CH5F3L 68324545 IC50 = 8210 nM T89534 C7KM0T 68779769 IC50 = 3.1 nM T89534 CHVW02 69281197 EC50 = 75 nM T89534 C6XQM8 70140794 IC50 = 20 nM T89534 C5AY3Z 70261892 IC50 = 5490 nM T89534 CBM80I 70354859 EC50 = 26.9 nM T89534 C4NMI7 70681450 IC50 = 0.6 nM T89534 CID9L6 70681451 IC50 = 0.2 nM T89534 C6YL4K 70681621 EC50 = 2.8 nM T89534 CT85IV 70681622 EC50 = 110 nM T89534 CFD6Y8 70681623 EC50 = 1300 nM T89534 CMI8Q9 70681848 IC50 < 100000 nM T89534 CARO49 70685018 Ki = 14 nM T89534 CZC61P 70685893 EC50 = 2.2 nM T89534 C6G1AZ 70685894 EC50 = 14 nM T89534 CF4D0J 70685895 EC50 = 200 nM T89534 CI3RN7 70685896 EC50 = 12 nM T89534 CJ5Z4N 70686080 IC50 < 100000 nM T89534 CR0MB3 70688747 EC50 = 120 nM T89534 CLO8E7 70690044 EC50 = 110 nM T89534 CNOJ60 70690045 EC50 = 2000 nM T89534 COU7T5 70690046 EC50 = 1200 nM T89534 C1KFL5 70690047 EC50 = 3150 nM T89534 CGU65P 70690163 Ki = 2.4 nM T89534 CWGC38 70692196 EC50 = 0.14 nM T89534 CH92NS 70694259 EC50 = 1100 nM T89534 CLVB71 70694260 EC50 = 210 nM T89534 CTK9H2 70694261 EC50 = 27 nM T89534 CGOH19 70694262 EC50 = 770 nM T89534 CY7EL2 70694264 EC50 = 2250 nM T89534 CIRY65 70694390 Ki = 5.3 nM T89534 CSWT16 70696334 EC50 = 670 nM T89534 CP5QM9 70696352 EC50 = 9.2 nM T89534 CZ72LR 70696353 EC50 = 11000 nM T89534 C3PM4W 70696354 EC50 = 5500 nM T89534 CRKF46 71153846 IC50 = 32500 nM T89534 CUH71V 71239417 IC50 > 1000 nM T89534 CG24SA 71449116 IC50 = 0.97 nM T89534 CW0N5Y 71450112 EC50 = 16 nM T89534 CJ3R1C 71450113 EC50 = 0.84 nM T89534 CGWH69 71453711 EC50 = 60 nM T89534 CDV74Z 71453712 EC50 = 0.12 nM T89534 CVB70T 71453742 EC50 = 0.31 nM T89534 C59KRH 71453743 EC50 = 100 nM T89534 COPG39 71454424 EC50 = 400 nM T89534 CG5H6B 71454465 IC50 = 6000 nM T89534 C15HIA 71455440 EC50 = 1.6 nM T89534 CN76BF 71457218 EC50 = 0.4 nM T89534 C2J7BX 71457266 EC50 = 0.67 nM T89534 CUAD52 71457267 EC50 = 47 nM T89534 C8DOM0 71457268 EC50 = 15 nM T89534 C2TN5I 71458013 IC50 = 235 nM T89534 C71HUY 71459076 EC50 = 0.27 nM T89534 CR14YQ 71459915 IC50 = 1700 nM T89534 CUAG08 71460882 EC50 = 0.2 nM T89534 CN87JE 71462585 EC50 = 24 nM T89534 CYW34A 71519686 IC50 = 3000 nM T89534 C83YJF 71544946 IC50 > 5000 nM T89534 CT9Y5D 71549558 IC50 = 3300 nM T89534 C8ZX0F 71549573 IC50 = 7300 nM T89534 CZ8Y7O 71549829 IC50 = 6100 nM T89534 CPFL57 71549843 IC50 = 17000 nM T89534 CY8SP0 71549969 IC50 > 20000 nM T89534 CX6JR5 71550242 IC50 = 7900 nM T89534 C6WIA2 71550244 IC50 = 6300 nM T89534 CSHT69 71550657 IC50 > 5000 nM T89534 COTM69 71580895 IC50 = 0.3 nM T89534 C8L6YZ 71609799 IC50 = 0.2 nM T89534 CNJD68 71609989 IC50 = 0.1 nM T89534 CB0N4Z 71609990 IC50 = 0.2 nM T89534 C6BDX7 71610523 IC50 = 1.5 nM T89534 COZ7X9 71610524 IC50 = 0.7 nM T89534 CW93GB 71610797 IC50 = 1.4 nM T89534 CPL0O7 71624342 EC50 = 2180 nM T89534 C9S4KZ 71624466 EC50 = 470 nM T89534 CA7F2B 71624467 EC50 = 1910 nM T89534 CGT86N 71624573 EC50 = 120 nM T89534 C1RV0Q 71624574 EC50 = 45 nM T89534 C2CLE1 71624678 EC50 = 1060 nM T89534 CD23NV 71624679 EC50 = 563 nM T89534 C6NZH1 71624682 EC50 = 65900 nM T89534 COK59Y 71624683 EC50 = 1160 nM T89534 CN06AS 71624796 EC50 = 1520 nM T89534 CFW3R0 71624797 EC50 = 439 nM T89534 CT1KP7 71624798 EC50 = 447 nM T89534 C5Y9LF 71624799 EC50 = 101 nM T89534 CN7KA2 71624911 EC50 = 615 nM T89534 CCFP43 71624912 EC50 = 66 nM T89534 C2C0LQ 71624915 EC50 = 485 nM T89534 CSZA43 71625041 EC50 = 387 nM T89534 C2DFZ4 71625042 EC50 = 9 nM T89534 C81GMJ 71625046 EC50 = 3790 nM T89534 CSOI92 71625169 EC50 = 3890 nM T89534 C1PD9I 71625173 EC50 = 944 nM T89534 C1M9GW 71625174 EC50 = 3640 nM T89534 C5XEQ9 71625175 EC50 = 266 nM T89534 C0OY8P 71661130 EC50 = 48360 nM T89534 CM3N9E 71712303 IC50 = 110 nM T89534 CNRU01 71712304 IC50 = 98 nM T89534 C8EY6K 71714518 IC50 = 1279 nM T89534 CLM0A3 71714519 IC50 = 2900 nM T89534 C8JS5K 71746266 EC50 = 0.8 nM T89534 CHDT07 71746268 EC50 = 0.4 nM T89534 C94DQT 71746269 EC50 = 0.4 nM T89534 CL4YX3 71746650 EC50 = 1.1 nM T89534 C56PQM 71746830 EC50 = 1 nM T89534 CUBP37 71765043 IC50 = 248 nM T89534 C1UA2B 71765044 IC50 = 127 nM T89534 CGJ5X4 71812208 IC50 > 5000 nM T89534 CN9M7E 71817803 IC50 = 222 nM T89534 CW36SK 73057389 IC50 = 145 nM T89534 CIS0D4 73057390 IC50 = 92 nM T89534 C7WEA2 73057393 IC50 = 484 nM T89534 C1AUC0 73057394 EC50 = 221 nM T89534 CE58TN 73333597 IC50 = 3100 nM T89534 CY4W5Z 73333703 IC50 = 12700 nM T89534 CSF52H 73333825 IC50 = 3200 nM T89534 C2RLP9 73346567 IC50 = 64908.26 nM T89534 CK3RU8 73347518 IC50 = 29.7 nM T89534 CA60OG 73348058 IC50 < 100000 nM T89534 CPVB67 73348059 IC50 = 64908.26 nM T89534 C4XOW1 73348859 EC50 = 12570 nM T89534 C5DTJ0 73350233 Ki = 190 nM T89534 CY53FM 73351956 EC50 = 8170 nM T89534 C1ZS5U 73352620 IC50 < 100000 nM T89534 CQN6M8 73353409 EC50 = 2550 nM T89534 C0G1IK 73353410 EC50 = 8320 nM T89534 CW6D9R 73354127 IC50 < 100000 nM T89534 CDKC58 73355642 IC50 < 100000 nM T89534 C9WY3B 73386689 EC50 = 15 nM T89534 CB4Q3X 73671443 EC50 = 6.2 nM T89534 CTVC21 73774965 EC50 = 61.5 nM T89534 C96JWC 73774966 EC50 = 5.2 nM T89534 C46ZFX 73775123 EC50 = 13.9 nM T89534 CK46UZ 73775278 EC50 = 5.3 nM T89534 C3L2WC 73775280 EC50 = 717.1 nM T89534 CCA4K2 74222430 EC50 = 0.8 nM T89534 CYGH56 76317236 IC50 = 14 nM T89534 CA9IX6 76328166 IC50 = 151 nM T89534 CP5E2V 76333018 EC50 = 7943.28 nM T89534 CX3T5H 76335417 IC50 = 100000 nM T89534 C0BF2I 76335716 IC50 = 26200 nM T89534 CA0D6H 76336630 EC50 = 31.62 nM T89534 C1B5KS 76336631 EC50 = 10000 nM T89534 C5KQ9A 77105904 IC50 = 0.4 nM T89534 C36YQX 78321756 IC50 = 23 nM T89534 CC90JF 78321758 IC50 = 78 nM T89534 CPH9Y0 78322066 IC50 = 4 nM T89534 CUD9B4 78322070 IC50 = 327 nM T89534 CELW49 78322377 IC50 = 316 nM T89534 CQ4B9L 78322379 IC50 = 31 nM T89534 C32SAW 78322380 IC50 = 647 nM T89534 C3FQG8 78322381 IC50 = 1 nM T89534 CLM34F 78322699 IC50 = 26 nM T89534 CEU36Z 78322700 IC50 = 941 nM T89534 CBHP24 78322701 IC50 = 886 nM T89534 C1G7VK 78322702 IC50 = 1030 nM T89534 CCP63W 78323006 IC50 = 1270 nM T89534 CBUP57 78323007 IC50 = 1823 nM T89534 CQMW35 78323008 IC50 = 26 nM T89534 CN2R0V 78323010 IC50 = 5020 nM T89534 CE09GU 78323328 IC50 = 1 nM T89534 C1MKR2 78323656 IC50 = 6 nM T89534 CG87TA 78323657 IC50 = 1 nM T89534 CNI07G 78323954 IC50 = 1 nM T89534 CY7DO8 78323955 IC50 = 58 nM T89534 C6Y5TP 78323956 IC50 = 40 nM T89534 C74MXP 78324253 IC50 = 55 nM T89534 C96CAJ 78324565 IC50 = 11 nM T89534 CZD3W9 78324876 IC50 = 17 nM T89534 C0ZE4D 78425809 EC50 = 2.1 nM T89534 CF3Q7K 86270891 EC50 = 0.6 nM T89534 C8J1FY 86270985 EC50 = 0.7 nM T89534 CRW92N 86270987 EC50 = 83 nM T89534 CIHS37 86270988 EC50 = 99 nM T89534 C7XPD4 86270989 EC50 = 1.8 nM T89534 CDJN45 86271086 EC50 = 37 nM T89534 C2VJ8M 86271087 EC50 = 7.4 nM T89534 CI9Y8M 86271089 EC50 = 1.7 nM T89534 CG79NV 86271184 EC50 = 17 nM T89534 CIF3C7 86271185 EC50 = 50 nM T89534 CA6PM4 86271186 EC50 = 28 nM T89534 CB5P2N 86271281 EC50 = 15 nM T89534 C8A1OX 86271282 EC50 = 300 nM T89534 CZ3D7B 86271283 EC50 = 90 nM T89534 CM83WK 86271284 EC50 = 12 nM T89534 C47MPR 86271285 EC50 = 190 nM T89534 CV0J7G 86271469 EC50 = 0.8 nM T89534 CA6J1C 86271471 EC50 = 1.1 nM T89534 CV90DA 86271553 EC50 = 1.6 nM T89534 CZ1N5T 86271645 EC50 = 4.2 nM T89534 C5KQ2Z 86271646 EC50 = 1.1 nM T89534 C5U6BO 86271738 EC50 = 5 nM T89534 C95BEZ 86271739 EC50 = 1.5 nM T89534 C1IZH2 86271742 EC50 = 1.9 nM T89534 C13XTI 86271833 EC50 = 0.8 nM T89534 CVQ71C 86271835 EC50 = 4.8 nM T89534 CHVL65 86271924 EC50 = 1.4 nM T89534 CP26ZM 86271925 EC50 = 2.8 nM T89534 CWN65V 86271926 EC50 = 4.1 nM T89534 CNEP10 86345430 IC50 = 1 nM T89534 C31WCG 86346166 IC50 = 0.1 nM T89534 CQRK65 86730685 IC50 = 3400 nM T89534 CTU83L 86763463 IC50 = 15 nM T89534 CB1VC0 86764136 IC50 = 0.4 nM T89534 CUJA92 86764241 IC50 = 0.2 nM T89534 C59GJF 87054925 IC50 = 13 nM T89534 C2U0BG 87055263 IC50 = 0.03 nM T89534 C5JK1L 89042295 IC50 = 112 nM T89534 CJSX36 89619690 IC50 = 0.2 nM T89534 CO07PH 89619977 IC50 = 0.1 nM T89534 C4O8HY 89634497 IC50 = 0.2 nM T89534 CB3I2O 89634514 IC50 = 11 nM T89534 CZH25C 89634609 IC50 = 0.1 nM T89534 CHVM10 89820253 EC50 = 4.3 nM T89534 CY6UE5 89820263 EC50 = 19 nM T89534 CJ0U4Y 89820264 EC50 = 0.3 nM T89534 CT3M7I 89820265 EC50 = 1.5 nM T89534 CMQ93G 90348277 IC50 > 10000 nM T89534 CF53CX 90372168 IC50 = 0.2 nM T89534 CK5F0Y 90372180 IC50 = 124 nM T89534 C5GFU4 90372433 IC50 = 5.4 nM T89534 CS3TR0 90372437 IC50 = 0.3 nM T89534 CVI17J 90372445 IC50 = 4.2 nM T89534 CK5D1A 90395281 IC50 = 17000 nM T89534 CK7MX2 90644079 EC50 = 0.3 nM T89534 C9S3GC 90644080 EC50 = 2.7 nM T89534 CB0QV8 90644081 EC50 = 20 nM T89534 C6YH5U 90644082 IC50 = 3 nM T89534 CEXC10 90644320 EC50 = 16 nM T89534 C1J2TA 90654352 IC50 = 26.2 nM T89534 COG3Q5 91668558 IC50 = 117 nM T89534 CYI89C 91810785 IC50 = 6.5 nM T89534 CU5XG6 102228006 IC50 = 10 nM T89534 CNJH98 102502192 EC50 = 96 nM T89534 C5ZR2C 102502193 EC50 = 61 nM T89534 CMO84S 110730849 IC50 = 204.75 nM T89534 C9FIG4 110730850 IC50 = 3.31 nM T89534 CIUL38 110730851 IC50 = 7.53 nM T89534 C6BDS9 112513964 IC50 = 69.46 nM T89534 C6VH5J 117094740 IC50 = 43 nM T89534 CNK71A 117611174 EC50 = 1.9 nM T89534 CX5FR2 117763076 IC50 = 0.3 nM T89534 CW27MY 118063735 EC50 > 10000 nM T89534 CI4GP9 118097391 EC50 > 10000 nM T89534 CQT2M7 118166573 IC50 = 1030 nM T89534 CU03DL 118166622 IC50 = 0.9 nM T89534 CB10GA 118166666 IC50 = 262 nM T89534 CF6MO1 118166678 IC50 = 7 nM T89534 CL5I0X 118166693 IC50 = 56 nM T89534 CV7ZG9 118166698 IC50 = 7 nM T89534 C7A8UH 118166720 IC50 = 113 nM T89534 CT0PZ7 118166734 IC50 = 0.8 nM T89534 CRTP56 118166740 IC50 = 120 nM T89534 CV2M7R 118166744 IC50 = 110 nM T89534 CH9QA7 118166788 IC50 = 219 nM T89534 CR32JE 118166789 IC50 = 2564 nM T89534 C7FD2S 118166792 IC50 = 112 nM T89534 C08UFT 118166812 IC50 = 1409 nM T89534 C24VKX 118166813 IC50 = 35 nM T89534 C96HPK 118166861 IC50 = 113 nM T89534 C69MNX 118184699 IC50 = 46 nM T89534 CBV6N0 118184700 IC50 = 1174 nM T89534 C06GNI 118184720 IC50 = 43 nM T89534 C7ZJR3 118184730 IC50 = 3 nM T89534 CQH23M 118184731 IC50 = 119 nM T89534 C0INJ8 118184735 IC50 = 15 nM T89534 C29NQM 118184739 IC50 = 5.5 nM T89534 CUG2Z0 118184741 IC50 = 0.6 nM T89534 CF6D0X 118184749 IC50 = 57 nM T89534 CRHI05 118184751 IC50 = 55 nM T89534 C5FC9X 118184760 IC50 = 15 nM T89534 CG69BK 118184761 IC50 = 77 nM T89534 CD1RJ8 118184777 IC50 = 0.4 nM T89534 C1Q8JO 118184782 IC50 = 27 nM T89534 CKLZ47 118184786 IC50 = 1.4 nM T89534 CC2YD0 118184807 IC50 = 207 nM T89534 C4LT7O 118184808 IC50 = 302 nM T89534 CK15YV 118184833 IC50 = 37500 nM T89534 CDK5I7 118184845 IC50 = 12 nM T89534 C4SBX9 118184846 IC50 = 139 nM T89534 CDKC49 118184849 IC50 = 505 nM T89534 C3JIB2 118184854 IC50 = 125 nM T89534 CIML42 118574931 IC50 = 216 nM T89534 CD3CK7 118574963 IC50 = 3 nM T89534 CLS7C1 118707978 Ki > 75000 nM T89534 C9LV0M 118707979 Ki > 75000 nM T89534 C6NIU0 118724546 IC50 = 13000 nM T89534 C3JU5H 118724548 IC50 = 230 nM T89534 C4UB8J 118724549 IC50 = 1100 nM T89534 CE0C6J 118724550 IC50 = 140 nM T89534 C7BRJ0 118724551 IC50 = 150 nM T89534 C5LR2N 118724552 IC50 = 40 nM T89534 CG1OL3 118724553 IC50 = 1470 nM T89534 CCK94J 118724554 IC50 = 18000 nM T89534 CW07TL 118724555 IC50 = 8 nM T89534 COJ81W 118735362 EC50 = 87.8 nM T89534 C8VFT2 118735363 EC50 = 277 nM T89534 CZE92I 118735364 EC50 = 274 nM T89534 CFB1G7 118735365 EC50 = 144 nM T89534 CX4V1E 118735366 EC50 = 1050 nM T89534 CW60ZD 118735367 EC50 = 675 nM T89534 C6ULM1 118735368 EC50 = 265 nM T89534 CE50LC 118735369 EC50 = 384 nM T89534 C6Y2NQ 118735371 EC50 = 653 nM T89534 C93CNO 118735374 EC50 = 290 nM T89534 C4YR6E 118735375 EC50 = 56.5 nM T89534 CS3ZJ8 118735376 EC50 = 176 nM T89534 CV83KA 118735377 EC50 = 3180 nM T89534 CG9RB4 118735379 EC50 = 34.9 nM T89534 CGT60X 118735380 EC50 = 27.1 nM T89534 CY6L8W 118735381 EC50 = 1920 nM T89534 C7VL3P 118737781 IC50 = 17 nM T89534 CQ4P8B 118737782 IC50 = 41 nM T89534 CZG3N7 118737783 IC50 = 5.9 nM T89534 CM14ON 118737784 IC50 = 9 nM T89534 C5XIC2 118737785 IC50 = 4.6 nM T89534 C5JTP6 118737786 IC50 = 1.6 nM T89534 C6V7AD 118737787 IC50 = 3 nM T89534 CJWX60 118737788 IC50 = 178 nM T89534 CC85BI 118737789 IC50 = 11 nM T89534 CES6O7 118737790 IC50 = 1.5 nM T89534 CNK32A 118737791 IC50 = 1 nM T89534 CUM9T0 118737792 IC50 = 256 nM T89534 CVN7J1 118737793 IC50 = 27 nM T89534 CVH7A9 118737794 IC50 = 0.5 nM T89534 CP4Y1L 118737795 IC50 = 25 nM T89534 CVM93U 118737796 IC50 = 9.9 nM T89534 C6N2PZ 118737797 IC50 = 1.3 nM T89534 CJN28K 118737798 IC50 = 7.4 nM T89534 C2XVQ5 118737799 IC50 = 3.2 nM T89534 C0MK1L 118737800 IC50 = 10 nM T89534 CZ8HX6 118737801 IC50 = 280 nM T89534 CT05AI 118737802 IC50 = 360 nM T89534 C6R2NI 118737803 IC50 = 100 nM T89534 CPA95Q 118737804 IC50 = 390 nM T89534 CBYP36 118737805 IC50 = 3600 nM T89534 CR6X9U 118737806 IC50 = 5800 nM T89534 CI53XV 118737807 IC50 = 330 nM T89534 C6E1WC 118737808 IC50 = 100 nM T89534 CIQ57L 118737845 IC50 = 50 nM T89534 CSJE19 118737846 IC50 = 50 nM T89534 C42PSU 118737847 IC50 = 1380 nM T89534 C8UP2N 121226004 IC50 = 55300 nM T89534 CWE9Y5 121241709 IC50 = 1.1 nM T89534 C0WO6T 121409920 IC50 = 0.58 nM T89534 CT0V7C 121409947 IC50 = 0.03 nM T89534 C68EUS 121409965 IC50 = 0.05 nM T89534 CP7N6H 121409995 IC50 = 0.2 nM T89534 C21AIE 121410016 IC50 = 3 nM T89534 CM2C0V 121410025 IC50 = 1 nM T89534 CZ68RS 121410042 IC50 = 0.5 nM T89534 C7CGK4 121410113 IC50 = 0.01 nM T89534 COS47H 121410578 IC50 = 0.07943 nM T89534 C8FN6J 121427080 IC50 = 0.045 nM T89534 CRUN70 121430327 IC50 = 0.5 nM T89534 CG13LX 122178361 IC50 = 4900 nM T89534 CT4Q1B 122178995 EC50 = 113 nM T89534 CVAY18 122178996 EC50 = 1050 nM T89534 CJ3LN0 122180153 IC50 = 53 nM T89534 C29JVK 122180154 IC50 = 3.6 nM T89534 C0TPU3 122180155 IC50 = 11 nM T89534 C8NQV0 122180156 IC50 = 4.8 nM T89534 C17TCM 122180157 IC50 = 210 nM T89534 C7QCB9 122180158 IC50 = 3.4 nM T89534 CRW9F3 122180812 Ki = 59.86 nM T89534 C3UO8M 122180813 EC50 = 1 nM T89534 CJ42OQ 122180814 Ki = 25 nM T89534 CRH37W 122180815 Ki = 56.57 nM T89534 CEW23B 122180816 Ki = 147.62 nM T89534 CBM0N2 122180817 Ki = 111.91 nM T89534 C7E2QD 122180818 Ki = 182.35 nM T89534 CBO5T8 122180819 Ki = 80.52 nM T89534 C3TB4Y 122180820 Ki = 2384.62 nM T89534 C3D4TV 122180821 EC50 = 1160 nM T89534 CC80JD 122180822 Ki = 104.02 nM T89534 CXPG14 122180823 Ki = 81.36 nM T89534 CS4OH2 122180824 Ki = 133.05 nM T89534 CB7MD5 122180825 EC50 = 16 nM T89534 CB51GT 122180826 Ki = 92.26 nM T89534 C1YZ6A 122180827 IC50 = 140 nM T89534 CYCT17 122180828 Ki = 126.02 nM T89534 COM0C9 122180829 Ki = 125.51 nM T89534 CP5ND8 122180830 IC50 = 790 nM T89534 CTPJ86 122180831 IC50 = 640 nM T89534 C4FJ1W 122180832 EC50 = 320 nM T89534 CF71OE 122180833 Ki = 121.57 nM T89534 CL16JS 122180834 Ki = 169.4 nM T89534 CE2A5S 122180835 Ki > 5000 nM T89534 CBC6D3 122181041 Ki > 5000 nM T89534 CP4ZJ2 122181042 Ki = 4428.57 nM T89534 COEZ74 122181043 Ki > 5000 nM T89534 C0EHV1 122181044 Ki > 5000 nM T89534 CA0KZ7 122181045 Ki > 5000 nM T89534 CE4AO3 122181046 EC50 = 1140 nM T89534 C7XP2A 122181047 Ki > 5000 nM T89534 CYD03G 122181048 IC50 = 160 nM T89534 C7QS2U 122183657 IC50 = 35 nM T89534 CF4V1K 122183658 IC50 = 13 nM T89534 C3KTX1 122183659 IC50 > 1000 nM T89534 CWB39X 122183660 IC50 = 620 nM T89534 C6XR8T 122183661 IC50 = 670 nM T89534 C2JPF0 122183662 IC50 > 1000 nM T89534 CH96CM 122183664 IC50 = 110 nM T89534 CBYI87 122183665 IC50 > 1000 nM T89534 CRUD13 122183666 IC50 > 1000 nM T89534 C1ZU3J 122183667 IC50 = 749 nM T89534 CXM1S6 122183668 IC50 = 94 nM T89534 CQ5IZ1 122183669 IC50 > 1000 nM T89534 C8QO1G 122183672 IC50 > 1000 nM T89534 CTX29Y 122183673 IC50 > 1000 nM T89534 CGJU04 122191773 IC50 = 3100 nM T89534 C0CLX7 122191774 IC50 = 24600 nM T89534 CN9C2T 122192181 IC50 = 1174.9 nM T89534 C80TIN 122192182 IC50 = 3715.35 nM T89534 CZG5N9 122192183 IC50 = 39.81 nM T89534 CBE26N 122192184 IC50 = 776.25 nM T89534 CP5ER0 122192185 IC50 = 43.65 nM T89534 CAR2M7 122192186 IC50 = 30.2 nM T89534 CZMK47 122192187 IC50 = 691.83 nM T89534 CCP56N 122192188 IC50 = 69.18 nM T89534 C3KH0N 122192189 IC50 = 97.72 nM T89534 CI8KN0 122192190 IC50 = 6.457 nM T89534 C95FVG 122192191 IC50 = 0.4169 nM T89534 C0T5CD 122620887 IC50 = 0.059 nM T89534 C7PUB4 122621200 IC50 = 0.055 nM T89534 CK08DJ 122621381 IC50 = 0.076 nM T89534 CP17KA 122622110 IC50 = 0.051 nM T89534 C4P9NG 122700657 EC50 = 289 nM T89534 C6CA4O 124088406 EC50 = 99 nM T89534 CNH4A8 124088429 EC50 > 10000 nM T89534 CEK31I 124148318 IC50 = 0.2512 nM T89534 C9QF2H 124222742 IC50 = 34 nM T89534 CF05QT 126480615 IC50 = 4.1 nM T89534 C94TWG 127025760 EC50 = 0.22 nM T89534 CEN47V 127029860 IC50 = 34.5 nM T89534 CCK36V 127029882 IC50 > 40000 nM T89534 CFY1P0 127029884 IC50 > 2000 nM T89534 C4M8QN 127030254 IC50 = 0.8 nM T89534 CCD7S3 127030255 IC50 = 0.4 nM T89534 CJQ73M 127030543 IC50 = 36 nM T89534 CQPR75 127030544 IC50 = 0.96 nM T89534 C3AFS4 127030545 IC50 = 3.981 nM T89534 CN5XW9 127030559 IC50 = 590 nM T89534 C47AYI 127030560 IC50 = 960 nM T89534 CZG9X5 127030821 IC50 = 82 nM T89534 CLDC46 127031152 IC50 > 37000 nM T89534 C60SMC 127031153 IC50 > 12000 nM T89534 CX4W7N 127031748 IC50 = 12.4 nM T89534 C1NYI0 127031749 IC50 = 81 nM T89534 C6W1YO 127032311 IC50 = 1.2 nM T89534 C4BXE0 127032365 IC50 = 1.7 nM T89534 CHAY10 127032366 IC50 = 1.6 nM T89534 CSN4B7 127032367 IC50 = 7.5 nM T89534 C2SGB4 127032368 IC50 = 1.3 nM T89534 CU0XT5 127032369 IC50 = 0.69 nM T89534 CR24LG 127032671 IC50 = 2.2 nM T89534 C2J4VF 127033264 IC50 = 5.8 nM T89534 CL7R1I 127033595 IC50 = 160 nM T89534 C39DUH 127033596 IC50 = 0.4 nM T89534 C7ZMR6 127033597 IC50 = 1.3 nM T89534 C9D2LE 127033598 IC50 = 0.25 nM T89534 C74SAW 127033892 IC50 = 22 nM T89534 CSV67L 127033893 IC50 = 31.9 nM T89534 C3QCS2 127033894 IC50 = 7.7 nM T89534 C3SR7L 127033895 IC50 = 27.1 nM T89534 CFI4S3 127033896 IC50 = 48.4 nM T89534 CF70TI 127034151 IC50 = 42 nM T89534 C12NMV 127034152 IC50 = 11 nM T89534 CLR2J7 127034153 IC50 = 1.3 nM T89534 CJK82T 127034154 IC50 = 5.5 nM T89534 C6HEU2 127034384 IC50 = 33.3 nM T89534 C0ZNT8 127034418 IC50 = 7 nM T89534 CEO3L9 127034419 IC50 = 170 nM T89534 CC6FD8 127034721 IC50 = 1060 nM T89534 C4EH3T 127034722 IC50 = 210 nM T89534 C2YXR7 127034902 IC50 = 2100 nM T89534 C9ZF0D 127035369 IC50 = 50 nM T89534 CLYC28 127038229 EC50 = 0.2 nM T89534 CUI43M 127041633 EC50 = 121 nM T89534 C1JEB2 127041634 EC50 = 436.2 nM T89534 CFB6K2 127042277 EC50 = 1 nM T89534 CWX5L7 127042278 EC50 = 58.7 nM T89534 C3G5TE 127042279 EC50 = 76.1 nM T89534 C0ZWQ9 127042604 EC50 = 30.6 nM T89534 C6JMT9 127042633 EC50 = 36.8 nM T89534 CEQ91U 127042898 EC50 = 18.5 nM T89534 CA0J4Q 127042930 EC50 = 33.4 nM T89534 CYU8Z5 127043892 IC50 = 18700 nM T89534 CHL5V4 127044059 IC50 = 17700 nM T89534 CV0Q2X 127044060 IC50 = 24900 nM T89534 C9S8CB 127044061 IC50 > 100000 nM T89534 C3SMP8 127045121 IC50 = 3400 nM T89534 CS04DH 127045122 IC50 = 19800 nM T89534 C5HFJ1 127045123 IC50 = 10600 nM T89534 C38BJS 127045271 IC50 > 100000 nM T89534 CF8R9C 127045272 IC50 = 35200 nM T89534 CSQ06E 127045273 IC50 = 6700 nM T89534 CC6W0E 127045274 IC50 = 7200 nM T89534 C9O4RK 127045434 IC50 = 23300 nM T89534 C8PZU3 127045576 IC50 = 39400 nM T89534 CQT56U 127045577 IC50 = 39800 nM T89534 CXK2T9 127045578 IC50 = 40300 nM T89534 CZ6O4S 127045579 IC50 = 38300 nM T89534 CT1Y6M 127049191 IC50 = 40 nM T89534 C24TMQ 127049192 IC50 = 0.09 nM T89534 C7B2GI 127049193 IC50 = 28 nM T89534 C3Q9UY 127049194 IC50 = 11 nM T89534 CZS07N 127049269 IC50 = 574 nM T89534 CLZR97 127049518 IC50 = 1.8 nM T89534 C4ITS1 127050198 IC50 = 380 nM T89534 CQ76OF 127050449 IC50 = 49 nM T89534 C2REL0 127051417 IC50 = 436 nM T89534 CBF64U 127051803 IC50 = 9 nM T89534 C12WOQ 129137247 EC50 = 72.1 nM T89534 CJB4M3 129137266 EC50 = 11036 nM T89534 CJ1N2M 129137280 EC50 = 212.9 nM T89534 CH42QX 129137285 EC50 = 1711 nM T89534 CZSB45 129205486 Ki = 0.65 nM T89534 CT61ZX 129205487 EC50 = 1.1 nM T89534 CV72WR 129205492 Ki = 0.5 nM T89534 CLRO76 129205499 EC50 = 0.07 nM T89534 C6G7VA 129205523 EC50 = 0.65 nM T89534 C1P3FN 129205616 EC50 = 0.24 nM T89534 C3OP0R 130232322 IC50 = 0.2 nM T89534 CG7T9C 130232326 EC50 = 0.2 nM T89534 CD1K0J 130232334 EC50 = 0.7 nM T89534 C75HQC 130232370 EC50 = 8 nM T89534 C1QY3W 130232392 IC50 = 67 nM T89534 C1EC2X 130232400 EC50 = 0.5 nM T89534 CO9A4K 130232401 EC50 = 1.5 nM T89534 CX1U6G 130232404 EC50 = 0.2 nM T89534 C70GWU 130232413 EC50 = 0.7 nM T89534 CRYS10 130232754 EC50 = 0.9 nM T89534 CG8WO3 130232762 IC50 = 0.2 nM T89534 CMX1V2 130232769 EC50 = 2 nM T89534 CP48SA 130232781 EC50 = 0.3 nM T89534 CR4D5M 130232807 EC50 = 0.5 nM T89534 C9GK1L 130232819 EC50 = 0.2 nM T89534 C3J5LN 130232873 EC50 = 1 nM T89534 C9JL4N 130232895 EC50 = 0.5 nM T89534 CI54NM 130232938 EC50 = 3 nM T89534 CF64WI 130232950 IC50 = 0.2 nM T89534 C57ASV 130232954 EC50 = 0.5 nM T89534 COJP50 130233149 EC50 = 2 nM T89534 CJ3UG9 130233175 IC50 = 38 nM T89534 CGZP38 130233179 IC50 = 0.7 nM T89534 C01ZBV 130233184 EC50 = 8 nM T89534 CEGJ04 130233196 EC50 = 0.3 nM T89534 CH5FI9 130233199 EC50 = 0.4 nM T89534 CKAC59 130233229 IC50 = 0.3 nM T89534 CD81EO 130233396 EC50 = 0.7 nM T89534 CN4RF6 132019596 IC50 = 0.3981 nM T89534 C0J4PZ 132046120 IC50 = 0.3981 nM T89534 CFUG87 132046174 IC50 = 0.631 nM T89534 CE9BL3 132046817 IC50 = 1 nM T89534 C32MHI 132046819 IC50 = 0.1995 nM T89534 CW8CI4 132046902 IC50 = 2.512 nM T89534 C5Y3MB 132502976 IC50 = 12 nM T89534 C79GMJ 132578496 IC50 > 10000 nM T89534 CWQK97 134130451 IC50 = 210 nM T89534 C74WMB 134133952 IC50 = 97 nM T89534 C2URL4 134134246 IC50 = 990 nM T89534 CD7NA5 134138492 IC50 = 2000 nM T89534 CCVJ27 134141761 IC50 = 86 nM T89534 CN7GJ2 134143539 IC50 > 10000 nM T89534 CP04WC 134144077 IC50 = 1700 nM T89534 CQO2G7 134148719 IC50 > 10000 nM T89534 CM8NP0 134149281 IC50 = 553 nM T89534 CFBX89 134149623 IC50 = 224 nM T89534 CYG76M 134150509 IC50 = 3340 nM T89534 C89SMK 134152807 IC50 > 10000 nM T89534 C1O0IW 134153257 IC50 > 10000 nM T89534 CK1BE9 134155077 EC50 = 451.2 nM T89534 C0Z4OD 134155524 IC50 = 875 nM T89534 C2BK3Z 134155779 EC50 = 164.1 nM T89534 C58OUX 134155994 IC50 = 20 nM T89534 CE08RT 134521164 EC50 = 0.3 nM T89534 CX53IF 134610856 IC50 = 10 nM T89534 C31BDG 134822336 IC50 = 195 nM T89534 C1G9FD 135348960 EC50 > 10000 nM T89534 C42PVJ 135400902 IC50 = 65 nM T89534 CL51KF 135400937 IC50 = 49 nM T89534 CBRN70 135400938 IC50 = 33 nM T89534 CY2GJ3 135401184 IC50 = 1500 nM T89534 CLX32H 135409570 Ki = 51 nM T89534 C6S5RV 135409748 IC50 = 246 nM T89534 CY39LP 135409961 IC50 = 1750 nM T89534 CO95DR 135409966 IC50 = 474 nM T89534 CMQE75 135412817 IC50 = 183 nM T89534 C1VWL3 135415992 IC50 = 7827 nM T89534 CPC1Q3 135421346 Ki = 25.12 nM T89534 CLN16H 135423261 IC50 = 47 nM T89534 C3BU7D 135423323 Ki = 7.943 nM T89534 CCRX48 135424620 IC50 = 98 nM T89534 CP9JN3 135424801 IC50 = 27569 nM T89534 C0KIP8 135425149 IC50 = 1753 nM T89534 CV2WX8 135428120 IC50 = 3 nM T89534 CXNV83 135430308 IC50 = 411 nM T89534 C30QWY 135430315 IC50 = 455 nM T89534 CK2ZF0 135431815 IC50 > 5000 nM T89534 CYJ7R0 135432882 IC50 = 8.5 nM T89534 CWCV13 135433141 Ki = 450 nM T89534 CA1MC6 135433906 IC50 = 30 nM T89534 CCI27T 135433989 IC50 = 196 nM T89534 CW7MZ8 135436561 IC50 > 5000 nM T89534 CAY0S9 135436566 IC50 = 4820 nM T89534 CCR8P7 135438141 IC50 = 475 nM T89534 C43PRB 135438183 EC50 = 3070 nM T89534 CC29NQ 135438201 IC50 = 463 nM T89534 CDA4B8 135438473 IC50 = 2260 nM T89534 CUXH34 135440385 Ki = 15.85 nM T89534 CBGO63 135443283 IC50 = 555 nM T89534 C8VWH0 135443287 IC50 = 5000 nM T89534 CX1T4W 135443301 IC50 = 1210 nM T89534 C21VTE 135445165 Ki = 125.89 nM T89534 CE50DW 135445365 IC50 = 1010 nM T89534 C60OGT 135445374 IC50 = 1340 nM T89534 CVM0P7 135446139 IC50 = 2854 nM T89534 CTD6A7 135449071 IC50 = 511 nM T89534 C78GFC 135454762 IC50 = 622 nM T89534 C9GZ1Q 135454811 IC50 = 1815 nM T89534 CEQ5F4 135457031 IC50 > 5000 nM T89534 C9BVI8 135457325 IC50 = 260 nM T89534 C2O1MP 135457889 Ki = 26 nM T89534 C1Z4BN 135458008 IC50 = 13 nM T89534 CCVE26 135458128 IC50 = 1309 nM T89534 CXU79B 135458129 IC50 = 3138 nM T89534 CY8U6E 135459005 IC50 > 100000 nM T89534 CHU54B 135461939 IC50 = 9620 nM T89534 CEB1W8 135471179 IC50 > 5000 nM T89534 CPO9D1 135477943 IC50 = 283 nM T89534 C17LIP 135481146 IC50 = 1435 nM T89534 C4O7RZ 135481158 IC50 > 10000 nM T89534 C8SE4C 135483639 IC50 = 2975 nM T89534 C6V1JZ 135483640 IC50 = 44 nM T89534 C6DI2R 135483660 IC50 = 1036 nM T89534 C0WP9D 135486163 EC50 = 901 nM T89534 CH9OV8 135487481 IC50 = 3080 nM T89534 CFO4V6 135489088 IC50 = 1047 nM T89534 CQ91HA 135489089 IC50 = 385 nM T89534 CAU4W8 135489212 Ki = 3162.28 nM T89534 CXY1Z2 135492323 IC50 = 431 nM T89534 CL5WG2 135492495 EC50 = 140 nM T89534 CMB9Z7 135493223 IC50 = 1813 nM T89534 CL20ZX 135494500 IC50 = 410 nM T89534 CTN2D6 135495080 IC50 = 227 nM T89534 CX3O9M 135495087 IC50 = 4040 nM T89534 CFDO01 135496191 IC50 = 1870 nM T89534 CB9Q3X 135496242 Ki = 10 nM T89534 CMK68Q 135497123 IC50 = 803 nM T89534 C90ZNW 135497128 Ki = 10 nM T89534 C2O8MY 135499764 IC50 = 717 nM T89534 CI09WX 135499787 IC50 = 3370 nM T89534 CE1D4V 135499837 IC50 = 2668 nM T89534 C3N9DF 135499972 IC50 = 443 nM T89534 CZ5Y9F 135500018 IC50 = 50 nM T89534 C25GWU 135500024 IC50 = 360 nM T89534 CRYW41 135502641 IC50 = 1100 nM T89534 C1RW9U 135503521 IC50 = 68 nM T89534 COF53G 135507181 Ki = 160 nM T89534 C67JAI 135507439 IC50 = 20 nM T89534 CPZ29O 135508382 IC50 = 163 nM T89534 C2ME7Q 135508383 IC50 = 809 nM T89534 C9GM1V 135508397 IC50 = 1980 nM T89534 CHO9X5 135508451 IC50 = 15 nM T89534 CFMN96 135511852 EC50 = 59 nM T89534 CJ60KF 135511863 EC50 = 1217 nM T89534 C7PZI5 135511869 IC50 = 2636 nM T89534 C9DZ7C 135511925 IC50 = 96 nM T89534 C67GSY 135511929 EC50 = 4790 nM T89534 CR7X1H 135511945 EC50 = 149 nM T89534 C61NSW 135514474 Ki = 100 nM T89534 CV6B8P 135515561 Ki = 20 nM T89534 C4XD9K 135516685 IC50 = 50 nM T89534 CGM5C6 135516694 IC50 = 6 nM T89534 CZKC69 135518123 IC50 = 24 nM T89534 CBPO32 135518124 IC50 = 1727 nM T89534 CVTD54 135518270 IC50 = 783 nM T89534 C3S5MX 135518313 IC50 = 559 nM T89534 CH6G0Q 135519304 IC50 = 4068 nM T89534 C3P8LZ 135519309 IC50 = 264 nM T89534 CU5J8M 135520120 IC50 = 48473 nM T89534 CR03JM 135522279 IC50 = 2638 nM T89534 C1OBI2 135524469 IC50 = 210 nM T89534 CNFZ03 135524510 EC50 = 549 nM T89534 CVX9H3 135524526 IC50 = 22 nM T89534 CMIE65 135524868 IC50 > 5000 nM T89534 C7TYU2 135524871 IC50 = 1030 nM T89534 C35TQU 135524884 IC50 = 59 nM T89534 CC46RN 135524945 Ki = 1584.89 nM T89534 CFQW27 135526994 IC50 = 273 nM T89534 CSZ1H7 135527005 EC50 = 140 nM T89534 CRKD27 135529495 Ki = 180 nM T89534 CQ0ZX7 135529496 Ki = 1260 nM T89534 CX1J8D 135535917 IC50 = 161 nM T89534 C15FTQ 135538030 IC50 = 138 nM T89534 CUCN57 135540445 IC50 = 1116 nM T89534 C84ZFX 135540483 IC50 = 31 nM T89534 CIKD94 135545359 IC50 = 249 nM T89534 C7X2CE 135547714 Ki = 7 nM T89534 CK7UM1 135547715 Ki = 47 nM T89534 C34JMK 135571931 IC50 > 100000 nM T89534 C4ODC2 135678114 Ki = 3333 nM T89534 CM0LN8 135817419 IC50 = 1 nM T89534 CSO3C1 135857090 IC50 = 1000 nM T89534 CED1L7 135871534 IC50 < 100000 nM T89534 CSY5I0 135871535 IC50 < 100000 nM T89534 CDJ1L6 135914665 EC50 > 100000 nM T89534 CALV45 135976649 Ki = 4200 nM T89534 CMJ41H 135987657 Ki = 490 nM T89534 CO0UC2 135987660 Ki = 2000 nM T89534 CP96SU 135987662 Ki = 210 nM T89534 C3I8VE 135987663 Ki = 650 nM T89534 CDG17Y 135987664 Ki > 3000 nM T89534 C9ABZ6 135987665 Ki = 130 nM T89534 C7GU8Q 135987666 Ki = 830 nM T89534 C4G1DL 135987668 Ki = 660 nM T89534 CIG6T5 135987670 Ki = 380 nM T89534 C1TV3R 135987671 Ki = 620 nM T89534 CSB76X 135987672 Ki = 70 nM T89534 C5B8SX 136002646 IC50 = 5100 nM T89534 C98FXW 136046127 EC50 = 3 nM T89534 CUN8F1 136046128 EC50 = 7 nM T89534 CX2KM3 136046129 EC50 = 5 nM T89534 CSOR78 136046131 EC50 = 1 nM T89534 CB1L2D 136046132 EC50 = 10 nM T89534 CQTA24 136046133 EC50 = 2 nM T89534 CB6YN3 136046134 EC50 = 23 nM T89534 CJ7AO4 136046135 EC50 = 2 nM T89534 C68OIK 136046136 EC50 = 1 nM T89534 CQ7K2A 136046137 EC50 = 14 nM T89534 CSCP10 136046138 EC50 = 7 nM T89534 C9LMN8 136046140 EC50 = 14 nM T89534 CJSU38 136046141 EC50 = 16 nM T89534 CU18VS 136046142 EC50 = 0.1 nM T89534 C5ORA9 136046143 EC50 = 15 nM T89534 CFGU03 136046144 EC50 = 4 nM T89534 CJ8X1O 136046145 EC50 = 57 nM T89534 C4P2BT 136046146 EC50 = 10 nM T89534 CXTR87 136046147 EC50 = 9 nM T89534 C9BI5M 136046148 EC50 = 7 nM T89534 CAH5S3 136046149 EC50 = 17 nM T89534 C0YZM4 136048726 IC50 = 376 nM T89534 CMI3Z2 136048727 IC50 = 196 nM T89534 C1BE8P 136048728 IC50 = 539 nM T89534 CRVT63 136048730 IC50 = 4652 nM T89534 CZG20O 136053633 EC50 = 64 nM T89534 CJC8N5 136053634 EC50 = 6900 nM T89534 CV3TP6 136053635 EC50 = 1400 nM T89534 CNW6H0 136053636 EC50 = 1700 nM T89534 C5WTV7 136053637 EC50 = 170 nM T89534 CRBK35 136053638 EC50 = 170 nM T89534 CRV6U5 136053639 EC50 = 46 nM T89534 C54YLG 136053640 EC50 = 12000 nM T89534 CCB5P6 136053641 EC50 = 1800 nM T89534 CO60LF 136053642 EC50 = 2000 nM T89534 CB54HV 136053643 EC50 = 900 nM T89534 CRA6C4 136053644 EC50 = 3100 nM T89534 CM35UY 136180341 EC50 = 29.3 nM T89534 CXP07U 136180342 EC50 = 194 nM T89534 CO79XD 136213601 IC50 = 7750 nM T89534 CR0ND2 136213603 IC50 = 1 nM T89534 CM9D8R 136213604 IC50 = 3 nM T89534 CVY5F4 136244610 IC50 < 100000 nM T89534 C38YOM 136260557 IC50 < 100000 nM T89534 C5GWA9 136497898 IC50 = 219 nM T89534 CKJ2F4 137175229 EC50 = 75 nM T89534 CC1XZ2 137175230 EC50 = 46 nM T89534 CM6EA1 137175231 EC50 = 77 nM T89534 CGH34U 137194225 EC50 = 0.2 nM T89534 C4HRL1 137503296 IC50 = 0.955 nM T89534 C4X2UQ 137503299 IC50 = 1.23 nM T89534 C5O4IG 137503303 IC50 = 1.023 nM T89534 C5IMN2 137503342 IC50 = 2.7 nM T89534 CC98EO 137503344 IC50 = 1.445 nM T89534 CZ90FS 137503669 IC50 = 1.413 nM T89534 CNXJ86 137628681 IC50 = 1943 nM T89534 CG79XQ 137631712 IC50 = 3510 nM T89534 CC64EG 137633461 Ki = 1.4 nM T89534 C2B3GJ 137634109 Ki = 0.13 nM T89534 CT03AC 137634796 Ki = 0.37 nM T89534 CMN0U2 137635165 IC50 = 63.2 nM T89534 CZ3V1F 137635423 Ki = 0.43 nM T89534 CIAM46 137637216 Ki = 0.18 nM T89534 C8OJ0I 137638372 Ki = 1.1 nM T89534 C2N3FX 137638822 IC50 = 1681 nM T89534 CP2VE3 137638954 IC50 = 2650 nM T89534 C85UAK 137639567 Ki = 0.35 nM T89534 CJV72U 137639609 Ki = 7.1 nM T89534 C9T6JB 137639849 IC50 = 6640 nM T89534 C32YMC 137640489 Ki = 0.57 nM T89534 CF8DG7 137640807 IC50 = 219 nM T89534 CLTS71 137641590 IC50 = 169 nM T89534 C8HP3M 137642810 Ki = 0.45 nM T89534 CRS0C8 137643006 IC50 = 294 nM T89534 CV5HA4 137643922 IC50 = 664 nM T89534 C5C9WQ 137645325 Ki = 3.3 nM T89534 CBY5H6 137645495 Ki = 0.71 nM T89534 C5Y2FO 137645971 IC50 = 10000 nM T89534 C2G3VI 137646525 Ki = 0.4 nM T89534 CHT21E 137646826 IC50 = 27 nM T89534 C9CWP1 137647667 Ki = 0.74 nM T89534 CX0JA8 137647962 Ki = 0.32 nM T89534 C5M7SV 137648055 IC50 = 158 nM T89534 CWP5O2 137649257 EC50 = 432 nM T89534 C8FVM1 137649725 IC50 = 1238 nM T89534 CE7K8L 137649825 Ki = 0.43 nM T89534 CNI49S 137650614 Ki = 0.37 nM T89534 C3O8KX 137651054 IC50 = 271 nM T89534 CR72HJ 137652183 Ki = 0.27 nM T89534 C2FZG3 137652281 IC50 = 1138 nM T89534 C8TR4J 137652311 IC50 > 10000 nM T89534 CWJ40L 137652508 IC50 = 154 nM T89534 CMR9Z4 137652975 IC50 = 1083 nM T89534 C1AS5K 137653286 IC50 = 9390 nM T89534 C57LME 137654397 Ki = 1.33 nM T89534 CMOA79 137656420 Ki = 0.36 nM T89534 CUPZ80 137657526 IC50 = 1654 nM T89534 C9LR5G 137658509 IC50 = 36 nM T89534 C7XP9V 137659010 Ki = 0.71 nM T89534 C40IML 137659097 Ki = 0.65 nM T89534 C1PE7V 137659936 Ki = 0.38 nM T89534 CN0SZ4 137660238 Ki = 0.37 nM T89534 C9FA3U 137660578 Ki = 1.7 nM T89534 CSQH43 137661589 IC50 = 225 nM T89534 CZ03SK 137661821 Ki = 0.71 nM T89534 CVY1M4 137662307 Ki = 1.8 nM T89534 CM3UF7 137700779 IC50 > 20000 nM T89534 CF1VR5 138693144 IC50 = 0.8 nM T89534 CC3E0R 138693215 IC50 = 0.5 nM T89534 C4U5PM 138693278 IC50 = 0.5 nM T89534 C01WKT 138693350 IC50 = 0.5 nM T89534 CPV1E4 138693568 IC50 = 0.6 nM T89534 CZ9E1A 139391843 IC50 = 2.1 nM T89534 CB0E1Y 139392008 IC50 = 8.128 nM T89534 CEO3I4 139392056 IC50 = 10.47 nM T89534 CA3I7J 139408644 IC50 = 5.129 nM T89534 CWKI95 139408668 IC50 = 12 nM T89534 C0K2JE 139408674 IC50 = 0.257 nM T89534 CPH0L4 139408675 IC50 = 1.905 nM T89534 CSXU49 139408681 IC50 = 3.02 nM T89534 CYS5L7 139408845 IC50 = 5.888 nM T89534 CMH90D 139408877 IC50 = 1.023 nM T89534 C6FJE2 139408939 IC50 = 5.2 nM T89534 CW2C4Z 139408951 IC50 = 0.5 nM T89534 CF8LN1 139582020 IC50 = 0.7943 nM T89534 CV26PQ 139582021 IC50 = 0.3981 nM T89534 CO05VM 145949224 IC50 = 539.18 nM T89534 CVC0B4 145950353 IC50 > 10000 nM T89534 CS05YB 145950468 IC50 = 5970 nM T89534 CZNX35 145951019 IC50 = 78 nM T89534 C4T0UE 145951407 IC50 > 10000 nM T89534 CHC8A3 145951614 IC50 > 10000 nM T89534 CWI7X0 145951633 IC50 = 168 nM T89534 CX9LI1 145951641 IC50 = 6430 nM T89534 CGSQ41 145952207 IC50 = 46.88 nM T89534 CRS3V5 145952243 IC50 > 10000 nM T89534 CGT02H 145953052 IC50 = 73.61 nM T89534 CJ86FH 145953150 IC50 = 8430 nM T89534 CG0YF8 145953184 IC50 = 80.36 nM T89534 C8WVA0 145953503 IC50 = 13200 nM T89534 CKP95X 145953707 IC50 > 10000 nM T89534 C97OLA 145953737 IC50 = 387.37 nM T89534 C2ZX1U 145953877 IC50 = 191.69 nM T89534 C65TWJ 145953883 IC50 > 10000 nM T89534 CCK17E 145953908 IC50 = 2190 nM T89534 CC7X6N 145953909 IC50 = 6870 nM T89534 CQ6N9J 145953976 IC50 = 3550 nM T89534 C7AUH9 145953977 IC50 > 10000 nM T89534 CX3BS8 145954021 IC50 = 6620 nM T89534 C8RA6E 145954397 IC50 = 4.9 nM T89534 CTV6X8 145954466 IC50 = 87 nM T89534 C3XOI2 145954572 IC50 = 3820 nM T89534 COK71C 145954893 IC50 = 6840 nM T89534 C0JNE2 145955665 IC50 = 4530 nM T89534 C6DK3T 145956091 IC50 = 16200 nM T89534 CM4W3N 145956205 IC50 = 259.16 nM T89534 CP69IC 145956222 IC50 = 60400 nM T89534 C1D4QT 145956476 IC50 = 4370 nM T89534 CN71VU 145956504 IC50 = 9420 nM T89534 CRN8U6 145956586 IC50 = 201.81 nM T89534 CO18XW 145957375 IC50 = 6430 nM T89534 CW21YS 145957522 IC50 = 78 nM T89534 C2Q5GH 145957892 IC50 = 33.13 nM T89534 CXU20C 145958661 IC50 = 76.73 nM T89534 CR58VX 145959073 IC50 = 300.43 nM T89534 C5IFM0 145959340 IC50 > 10000 nM T89534 CT0QR2 145959503 IC50 = 29400 nM T89534 CS0G2T 145959695 IC50 = 7790 nM T89534 C1WZ5V 145959741 IC50 = 8210 nM T89534 C5KOI6 145959948 IC50 > 200000 nM T89534 C7RK8L 145960186 IC50 = 4.9 nM T89534 C2X7DZ 145960328 IC50 = 7960 nM T89534 CKBW57 145960786 IC50 = 20 nM T89534 CKN29E 145961426 IC50 = 2620 nM T89534 C3U4RJ 145961651 IC50 > 10000 nM T89534 CCF02H 145964530 IC50 = 4100 nM T89534 C56SHA 145964597 IC50 = 4700 nM T89534 CMG6W2 145964616 Ki = 107.38 nM T89534 CVJ7L6 145964633 Ki = 62.1 nM T89534 C8QI0U 145965134 Ki = 51.32 nM T89534 CHF39D 145965184 IC50 = 55000 nM T89534 C9A3UM 145965217 IC50 = 2 nM T89534 C5H8EZ 145965425 IC50 = 1700 nM T89534 C2T3PU 145965787 IC50 = 0.5 nM T89534 CM9LG0 145965903 Ki = 168.6 nM T89534 C8K1WV 145965925 Ki = 153.07 nM T89534 CA6CZ4 145966389 IC50 = 19 nM T89534 CS9MD6 145966668 Ki = 129.74 nM T89534 C0WG5H 145966819 Ki = 498.57 nM T89534 CU4MD5 145967018 IC50 = 26640 nM T89534 CE4S7F 145967279 IC50 = 48 nM T89534 CNJO46 145967622 IC50 = 57 nM T89534 C80AGW 145967704 IC50 = 59 nM T89534 CB68HI 145967819 IC50 = 22440 nM T89534 C8KNI7 145967847 IC50 = 429 nM T89534 C8H3YV 145968201 IC50 = 71.6 nM T89534 C8VQ5G 145968272 IC50 > 10000 nM T89534 C1S0TJ 145968278 IC50 = 4.1 nM T89534 CXN86W 145968289 IC50 = 349 nM T89534 CE1WK0 145968307 IC50 = 634 nM T89534 C8BF1J 145968369 IC50 = 11.7 nM T89534 CRUO57 145968523 IC50 = 147 nM T89534 C2CE4P 145968537 IC50 = 104 nM T89534 CD86FU 145968562 IC50 = 1023 nM T89534 CY78XO 145968786 IC50 = 1040 nM T89534 C2DNL3 145968920 IC50 = 482300 nM T89534 CT8R7I 145968943 Ki = 249.29 nM T89534 CL6IQ4 145969020 IC50 = 613 nM T89534 C40OKG 145969029 IC50 > 10000 nM T89534 CEQ15L 145969388 IC50 = 60780 nM T89534 CY0VA4 145969440 IC50 = 14 nM T89534 C86AEM 145969473 IC50 = 1129 nM T89534 CO75XN 145969585 IC50 = 14 nM T89534 CEY2I5 145969791 IC50 = 21 nM T89534 C7PQH3 145969854 IC50 = 49 nM T89534 CXY0E1 145970107 IC50 = 74 nM T89534 CW1D3A 145970135 IC50 > 10000 nM T89534 C93BQD 145970491 IC50 = 61080 nM T89534 CVY9Q7 145971019 IC50 = 587190 nM T89534 CH0X7P 145971353 IC50 = 355790 nM T89534 CVW6D7 145972047 Ki = 240.69 nM T89534 C4KJX2 145972317 Ki = 634.55 nM T89534 CAVN67 145972459 IC50 = 4270 nM T89534 CLJ4Y7 145972474 IC50 > 10000 nM T89534 CQ47XM 145972475 IC50 > 10000 nM T89534 C1QF2L 145972690 IC50 = 2.4 nM T89534 CDQ7E0 145972963 Ki > 10000 nM T89534 C4OF2V 145973074 IC50 = 5 nM T89534 C5TP2F 145973118 IC50 = 400 nM T89534 CI6T9M 145973161 IC50 = 40 nM T89534 C37FBS 145973441 Ki = 251.08 nM T89534 CFKW97 145973654 IC50 = 18410 nM T89534 C3AZ4O 145973866 Ki = 29.7 nM T89534 CXZS64 145974009 IC50 = 10 nM T89534 CWC19X 145974551 IC50 > 10000 nM T89534 CJ62QA 145974791 IC50 = 8960 nM T89534 CQZ7D8 145975059 Ki = 40.77 nM T89534 CM01NE 145975361 IC50 = 2 nM T89534 C5V2AD 145975958 IC50 = 16550 nM T89534 C5MJ9W 145975973 IC50 = 3860 nM T89534 CE5N1B 145976228 IC50 = 54 nM T89534 C4Q9KI 145976280 IC50 = 61 nM T89534 CR0ON9 145976505 IC50 = 51190 nM T89534 C8DS5Q 145976853 Ki = 149.15 nM T89534 C4DPO7 145976892 EC50 = 4 nM T89534 CRJU43 145976968 Ki = 53.28 nM T89534 CO70FX 145977155 IC50 = 9270 nM T89534 C7IL3R 145977161 Ki = 10.51 nM T89534 CE75OD 145977494 EC50 = 18 nM T89534 CVX45W 145977605 IC50 = 62 nM T89534 C9MG6O 145977673 Ki = 43.03 nM T89534 C98CHS 145977976 IC50 = 5200 nM T89534 CKQ5C2 145978265 EC50 = 2 nM T89534 CS0N8E 145978277 IC50 = 3 nM T89534 C0D9ES 145978643 IC50 = 0.4 nM T89534 C43SYL 145978903 IC50 = 974 nM T89534 C1AJL5 145979357 EC50 = 116 nM T89534 CCBN24 145979638 IC50 = 415 nM T89534 CE80KP 145980527 IC50 = 874 nM T89534 CJ5U0Y 145980901 EC50 = 136 nM T89534 CLJ3S7 145981530 IC50 = 13 nM T89534 CVC58M 145981549 EC50 = 911 nM T89534 C21SIT 145981553 IC50 = 69 nM T89534 CSM61H 145981867 IC50 = 1589 nM T89534 C7UH4A 145982555 IC50 = 5130 nM T89534 C9KR5H 145982571 IC50 = 2170 nM T89534 CY08OG 145982591 IC50 = 1120 nM T89534 C8UZV2 145982754 IC50 = 3420 nM T89534 CRT9I3 145982975 IC50 = 800 nM T89534 C10XYG 145983072 IC50 = 1200 nM T89534 CNOG85 145983259 IC50 = 1940 nM T89534 C0O1NY 145983278 IC50 = 2860 nM T89534 CCRI70 145983336 Ki = 25 nM T89534 CD69JB 145983784 IC50 = 10000 nM T89534 C05MBI 145983837 IC50 = 390 nM T89534 CP27UK 145983884 Ki = 11 nM T89534 CYZO43 145984038 Ki = 185 nM T89534 CYUD47 145984188 IC50 = 220 nM T89534 CVJY47 145984216 Ki = 0.07 nM T89534 CVH6Y9 145984234 IC50 = 5960 nM T89534 CY79IW 145984263 IC50 = 760 nM T89534 CQ9A0N 145984791 IC50 = 4740 nM T89534 CDM05I 145985073 IC50 = 80 nM T89534 C0O2AR 145985081 IC50 = 89 nM T89534 CEF7W4 145985090 IC50 = 1640 nM T89534 C9MV2L 145985198 IC50 = 820 nM T89534 CC3U1S 145985468 IC50 = 6220 nM T89534 CO50ZW 145985605 Ki = 1541 nM T89534 C3O4HE 145985821 Ki = 6.9 nM T89534 C31MIF 145985835 IC50 = 1800 nM T89534 CG8O2K 145986244 IC50 = 96 nM T89534 CN91YC 145986320 EC50 = 158 nM T89534 CF49OP 145986577 IC50 = 4677 nM T89534 CMQK52 145986591 IC50 = 23 nM T89534 C28LAH 145986759 IC50 = 769 nM T89534 CA1D2B 145987043 IC50 = 48 nM T89534 CPRH38 145987084 EC50 = 1003 nM T89534 CF9S0O 145987265 IC50 = 407 nM T89534 CKYW98 145988223 EC50 = 204 nM T89534 CK5RV0 145988666 EC50 > 10000 nM T89534 C09MNB 145988825 IC50 = 67 nM T89534 CW0C8Y 145989462 EC50 = 1831 nM T89534 CX74YQ 145989561 EC50 = 199 nM T89534 CSF03L 145989681 IC50 = 41 nM T89534 CR0LK9 145989755 EC50 = 721 nM T89534 COI2R8 145991129 EC50 = 219 nM T89534 C2NH3M 145991296 IC50 = 413 nM T89534 CP4V8N 145991796 IC50 = 179 nM T89534 CQ1WY2 146183836 IC50 = 0.79 nM T89534 C04KLS 146428237 IC50 = 0.24 nM T89534 C9K2RG 146428250 IC50 = 0.61 nM T89534 CWG2N1 146567341 IC50 = 0.7 nM T89534 CFNR34 146567342 IC50 = 0.49 nM T89534 C43PZX 146567347 IC50 = 0.37 nM T89534 C8ZL7B 146567366 IC50 = 0.82 nM T89534 CFD3E8 146567377 IC50 = 0.5 nM T89534 C5G2BR 146567380 IC50 = 0.3 nM T89534 C3C1XK 146567381 IC50 = 0.7 nM T89534 C46GUI 149822983 IC50 = 0.5 nM T89534 C6Y8BH 155510359 IC50 = 2980 nM T89534 CF8PO7 155511409 IC50 = 2.4 nM T89534 CCGY16 155511936 IC50 = 0.3162 nM T89534 C7VS5G 155511937 IC50 = 1240 nM T89534 CIJ4K9 155512714 IC50 = 27 nM T89534 CVCK17 155513135 IC50 > 10000 nM T89534 C2PU1J 155513315 IC50 = 1700 nM T89534 CGKQ42 155513962 IC50 = 0.021 nM T89534 CMQC26 155515404 IC50 = 1658 nM T89534 CP1L3J 155516697 IC50 > 10000 nM T89534 CL80FT 155516984 EC50 = 2 nM T89534 CFJO71 155518954 IC50 = 0.17 nM T89534 CLR23U 155519218 IC50 > 5000 nM T89534 CY94AM 155520303 IC50 = 90 nM T89534 C5CXT0 155520789 EC50 = 20 nM T89534 CMWI40 155521404 IC50 = 1780 nM T89534 C7LVS8 155521699 IC50 = 0.8 nM T89534 C4RK1P 155522067 IC50 = 15 nM T89534 C3LNK9 155522178 IC50 = 63.1 nM T89534 CSE31P 155522268 IC50 = 0.28 nM T89534 C9MAF1 155525071 IC50 = 0.42 nM T89534 C4PIM5 155526909 IC50 = 7.5 nM T89534 CAJW03 155527870 IC50 = 5.7 nM T89534 CSLJ15 155528850 IC50 > 10000 nM T89534 C0GY8X 155529068 IC50 = 0.7943 nM T89534 CUO74Y 155529729 EC50 = 0.6 nM T89534 CH42RB 155530321 IC50 = 0.07 nM T89534 CE4S3C 155533437 IC50 = 4.71 nM T89534 C0TW8H 155534195 IC50 = 94 nM T89534 CC5HJ6 155535796 IC50 > 10000 nM T89534 CI5T9E 155536687 EC50 = 1.3 nM T89534 CS06LK 155537645 EC50 = 140 nM T89534 CYS47I 155537918 IC50 > 100 nM T89534 C9EW1F 155538055 IC50 = 0.2 nM T89534 CH3V8J 155538711 EC50 = 427 nM T89534 CB3CY8 155538987 IC50 = 2500 nM T89534 COP7X8 155539171 IC50 > 10000 nM T89534 C4ID8Q 155539669 IC50 > 5000 nM T89534 CA2G8E 155539747 IC50 = 0.3162 nM T89534 C90XVB 155539810 IC50 = 25.12 nM T89534 CKF67H 155540121 IC50 = 1.995 nM T89534 C2RAP5 155540472 IC50 > 100 nM T89534 CMT91D 155540730 IC50 = 2300 nM T89534 C31CNR 155541121 IC50 > 5000 nM T89534 C8MPH9 155541236 IC50 = 1.259 nM T89534 CL53BE 155543769 IC50 = 2460 nM T89534 CU9A7M 155544127 Ki = 25 nM T89534 CF6TH5 155546055 IC50 = 2.5 nM T89534 CT0ON6 155546145 IC50 = 31 nM T89534 CP9Y8J 155548583 IC50 > 5000 nM T89534 C2PUT5 155549053 EC50 = 93 nM T89534 CA5G2T 155551013 IC50 > 10000 nM T89534 CRS02E 155551888 IC50 = 2330 nM T89534 CS9D3O 155552434 IC50 > 100 nM T89534 CF68WS 155552480 IC50 = 100 nM T89534 C5MHU4 155552943 IC50 > 5000 nM T89534 C1DC4A 155553793 IC50 = 30 nM T89534 C5S9LI 155556292 IC50 > 10000 nM T89534 CT3F5K 155556316 IC50 = 0.5 nM T89534 CY1S3T 155557113 IC50 = 8.15 nM T89534 C7AJZ5 155559268 IC50 = 1142 nM T89534 CHI07R 155559518 EC50 = 1 nM T89534 CLJ4A1 155559849 IC50 > 100 nM T89534 C2D6ZM 155561414 EC50 > 500 nM T89534 CV5I6E 155562017 IC50 = 37 nM T89534 C4CJ7W 155562234 IC50 = 250000 nM T89534 C9KY5I 155562382 IC50 > 10000 nM T89534 CSJQ98 155562658 IC50 = 22.67 nM T89534 C5NR7H 155562810 IC50 = 213 nM T89534 C48NOU 155563946 EC50 = 0.2 nM T89534 C7JMZ0 155564173 IC50 = 0.3 nM T89534 CQ97FI 155564996 IC50 = 72 nM T89534 CWK95R 155565459 IC50 > 10000 nM T89534 CY71WP 155565677 IC50 > 10000 nM T89534 C2UTY4 155566549 IC50 = 0.631 nM T89534 CT7OB2 155566794 IC50 = 19.95 nM T89534 C4C9PF 155566802 IC50 = 0.3162 nM T89534 C4HFX0 155566914 EC50 = 193 nM T89534 CMX67L 155567147 IC50 = 2116 nM T89534 C2NBO7 155567224 IC50 = 0.3 nM T89534 CY28HU 155567231 IC50 > 5000 nM T89534 C76EWQ 155567785 IC50 = 1.76 nM T89534 C4ZQ7D 155568522 IC50 = 1 nM T89534 CJRS26 155568547 IC50 = 6300 nM T89534 C4JTH2 155568868 IC50 > 5000 nM T89534 C5I0QV 155569431 IC50 = 0.08 nM T89534 CVD17E 10087534 EC50 = 380 nM T89534 C0RGJ9 44389594 EC50 = 1.1 nM T89534 D00CWN 135987619 Ki = 310 nM T89534 D00DJX 44597742 IC50 = 11 nM T89534 D00HZT 135449109 IC50 = 780 nM T89534 D00IXB 10445833 IC50 = 101 nM T89534 D00NEK 44405867 IC50 = 8310 nM T89534 D00RIX 5280443 IC50 = 1253 nM T89534 D00URP 10399473 IC50 = 1030 nM T89534 D00XLU 44407802 EC50 = 242 nM T89534 D00ZBL 135458122 IC50 = 727 nM T89534 D01AHL 44412953 IC50 > 10000 nM T89534 D01CYI 11579721 IC50 = 53640 nM T89534 D01GPY 10192794 IC50 = 40 nM T89534 D01IAT 10171410 IC50 = 2642 nM T89534 D01KJU 6102690 IC50 = 91 nM T89534 D01KSR 135495079 IC50 = 2765 nM T89534 D01QXL 9993627 IC50 = 153 nM T89534 D01SWO 9901869 IC50 = 35 nM T89534 D01TUB 135519319 IC50 = 213 nM T89534 D01WCA 656936 IC50 = 176 nM T89534 D01XCA 44407801 EC50 = 534 nM T89534 D02DML 5281707 IC50 = 11 nM T89534 D02EJM 136048731 IC50 = 775 nM T89534 D02GLM 9994500 Ki = 2800 nM T89534 D02HGS 135502634 IC50 = 632 nM T89534 D02JJU 135492380 IC50 = 3800 nM T89534 D02LCC 135442595 IC50 = 1200 nM T89534 D02OKF 10308197 IC50 = 10 nM T89534 D02RQP 6623 EC50 = 290 nM T89534 D02TPO 10323679 IC50 = 10 nM T89534 D02WRU 11201035 Ki = 2222 nM T89534 D02WSA 11579722 IC50 = 75588 nM T89534 D02XVV 10399376 IC50 > 10000 nM T89534 D02ZSX 61253 IC50 = 8740 nM T89534 D03BOO 25128804 Ki = 4100 nM T89534 D03CBX 135454802 IC50 = 212 nM T89534 D03DVM 10131379 IC50 = 31 nM T89534 D03GYS 135499774 IC50 = 498 nM T89534 D03NTD 9878556 Ki = 132 nM T89534 D03QHG 16066665 IC50 = 216 nM T89534 D03RYU 135522275 IC50 = 82 nM T89534 D03XEU 10286022 IC50 = 483 nM T89534 D04EAY 135474202 IC50 = 3000 nM T89534 D04SAO 9799518 EC50 = 1.7 nM T89534 D04TPC 25130896 Ki > 7300 nM T89534 D04WHH 135519317 IC50 = 390 nM T89534 D05EOW 102614 EC50 = 3.4 nM T89534 D05FUY 10149584 IC50 = 43 nM T89534 D05JKC 135546593 IC50 = 464 nM T89534 D05JPW 135409725 IC50 = 2557 nM T89534 D05KXP 44418726 IC50 = 1017 nM T89534 D05LQD 10082995 IC50 > 10000 nM T89534 D05PNP 11064571 IC50 = 26200 nM T89534 D05YIU 10236250 IC50 = 6.8 nM T89534 D06DDT 5315502 EC50 = 1590 nM T89534 D06OAL 135442585 IC50 = 537 nM T89534 D06SCS 135418373 IC50 = 155 nM T89534 D07HBQ 25128814 IC50 = 2400 nM T89534 D07LUI 11459006 IC50 = 211 nM T89534 D07TGS 3017674 IC50 = 150 nM T89534 D07TGW 135857091 IC50 = 20 nM T89534 D07VPM 135409756 IC50 = 1300 nM T89534 D07XBD 10308075 IC50 = 282 nM T89534 D07XUY 44418717 IC50 = 5245 nM T89534 D08FLV 135474625 IC50 = 819 nM T89534 D08GWS 46919124 Ki = 25.43 nM T89534 D08HCF 135496133 IC50 = 5000 nM T89534 D08LVT 44407806 IC50 = 1371 nM T89534 D08SJL 135524856 IC50 = 1500 nM T89534 D08VDX 10214699 IC50 = 30 nM T89534 D08WDN 135496123 IC50 = 6100 nM T89534 D09CQC 135471161 IC50 = 902 nM T89534 D09DEK 10171409 IC50 = 442 nM T89534 D09FWP 11368353 IC50 > 5000 nM T89534 D09FWS 135430317 IC50 = 634 nM T89534 D09NFD 6852176 IC50 = 320 nM T89534 D09NOH 44418728 IC50 = 140 nM T89534 D09PXU 9991961 IC50 = 4610 nM T89534 D09TQE 135528620 IC50 = 1570 nM T89534 D09ULU 2368773 IC50 = 404 nM T89534 D09UQU 10029432 IC50 = 64 nM T89534 D09UWI 14905189 EC50 = 2350 nM T89534 D09WEK 135503667 EC50 = 390 nM T89534 D0AD3U 135528621 IC50 = 8430 nM T89534 D0AD8G 44407887 IC50 = 235 nM T89534 D0AU0M 637542 EC50 = 16120 nM T89534 D0B1HP 135526958 IC50 = 815 nM T89534 D0C4VX 135407148 IC50 = 52 nM T89534 D0C5FY 10331951 IC50 = 654 nM T89534 D0C6AP 10285954 IC50 = 114 nM T89534 D0C6UR 49863610 Ki = 13.66 nM T89534 D0C9XK 135545334 IC50 = 2410 nM T89534 D0C9XW 11276767 IC50 = 13000 nM T89534 D0CC6R 10125290 IC50 = 24 nM T89534 D0D1LB 44418733 IC50 = 503 nM T89534 D0DK9S 135454786 IC50 = 6240 nM T89534 D0F1SS 44605900 EC50 > 10000 nM T89534 D0F8LS 135524867 IC50 = 18 nM T89534 D0FD6Z 10308090 IC50 = 22 nM T89534 D0H1CO 10244394 IC50 = 1880 nM T89534 D0H2FI 10308268 IC50 = 709 nM T89534 D0H5HI 9993278 IC50 = 468 nM T89534 D0H6MZ 25133613 IC50 = 7300 nM T89534 D0H8PI 10308021 IC50 = 22 nM T89534 D0H8ZT 135525228 IC50 = 37 nM T89534 D0HD2G 4788 IC50 = 300 nM T89534 D0HM8Y 44408971 IC50 = 1170 nM T89534 D0HR8L 11447703 IC50 = 1452 nM T89534 D0I1NX 10246180 EC50 = 0.15 nM T89534 D0I5HZ 44405888 IC50 = 1800 nM T89534 D0I5VJ 135520257 IC50 = 55883 nM T89534 D0J0AG 135421237 IC50 = 1140 nM T89534 D0J2NG 44418724 IC50 = 392 nM T89534 D0J3PM 44407886 EC50 = 1985 nM T89534 D0J6KN 135511848 IC50 = 40 nM T89534 D0K0IC 13896065 IC50 = 24 nM T89534 D0K0TR 11356877 IC50 1000000 nM T89534 D0K1TW 135443280 IC50 = 5280 nM T89534 D0K5LX 135566322 IC50 = 48 nM T89534 D0K6TE 10286087 IC50 = 107 nM T89534 D0K7HR 135409729 IC50 = 504 nM T89534 D0K8QD 63059 EC50 = 0.015 nM T89534 D0L0RK 44407885 EC50 = 1430 nM T89534 D0L2MU 10286352 IC50 = 1.5 nM T89534 D0L3AX 236868 IC50 = 638 nM T89534 D0L6IQ 135424609 IC50 = 6630 nM T89534 D0LI0M 44418723 IC50 = 383 nM T89534 D0M0RS 11560224 Ki > 1000 nM T89534 D0M0XL 11414445 IC50 = 884 nM T89534 D0M4LQ 44407804 EC50 = 705 nM T89534 D0MY8V 10308207 IC50 = 92 nM T89534 D0N0OY 135405741 IC50 = 1227 nM T89534 D0NN0V 637048 IC50 = 10200 nM T89534 D0O2KP 12133211 IC50 = 58 nM T89534 D0O5KR 10060956 IC50 = 335 nM T89534 D0O6FX 10061675 IC50 = 237 nM T89534 D0O9NE 5388063 Ki = 261 nM T89534 D0OV3S 11782482 IC50 = 50 nM T89534 D0P4SR 11716633 EC50 = 17 nM T89534 D0P6FN 10125342 IC50 = 174 nM T89534 D0P7PK 77020 IC50 = 6950 nM T89534 D0P8PK 10192730 IC50 = 230 nM T89534 D0Q4VG 135458016 IC50 = 25 nM T89534 D0Q6MS 11141183 IC50 = 30 nM T89534 D0R7AG 135486039 IC50 = 190 nM T89534 D0R7QY 127676 EC50 = 2600 nM T89534 D0S0SZ 135409723 IC50 = 481 nM T89534 D0S2ZJ 135430305 IC50 = 2353 nM T89534 D0S5RI 11547961 Ki = 13.01 nM T89534 D0S6NV 10149684 IC50 = 266 nM T89534 D0S8AV 509245 IC50 = 57 nM T89534 D0S8EB 11777167 IC50 = 1210 nM T89534 D0SR8Q 11458674 IC50 = 3405 nM T89534 D0SY2M 5281708 IC50 = 450 nM T89534 D0U0ZE 44408769 IC50 = 585 nM T89534 D0U2VA 4369550 IC50 = 117 nM T89534 D0U7KV 201385 IC50 = 94.8 nM T89534 D0UV9G 10125182 IC50 = 1345 nM T89534 D0V6KJ 10214708 IC50 = 10.3 nM T89534 D0V7OK 6366969 IC50 = 7 nM T89534 D0V7QZ 135528624 IC50 = 139 nM T89534 D0V7ZI 135476471 EC50 = 98 nM T89534 D0VN2R 10171886 IC50 = 1231 nM T89534 D0W0LG 44418722 IC50 = 155 nM T89534 D0W2YR 135522274 IC50 = 5110 nM T89534 D0W3FF 135503567 IC50 = 1900 nM T89534 D0W4WF 100801 IC50 = 240 nM T89534 D0W5HT 44418725 IC50 = 436 nM T89534 D0WM5O 5322399 Ki > 10000 nM T89534 D0WP6A 5348729 IC50 > 10000 nM T89534 D0X0RJ 9848809 IC50 = 76 nM T89534 D0X2VK 9945207 IC50 = 4.3 nM T89534 D0X4VN 10236221 IC50 = 92 nM T89534 D0X6LK 10823890 IC50 = 2700 nM T89534 D0X7DJ 10308206 IC50 = 27 nM T89534 D0X7SR 10246505 EC50 = 50 nM T89534 D0XC3V 10871661 IC50 = 500 nM T89534 D0XF9F 135484659 Ki = 2.7 nM T89534 D0XS0R 44433505 Ki > 1100 nM T89534 D0Y2LJ 44418729 IC50 = 80 nM T89534 D0Y4NJ 11784736 IC50 = 0.28 nM T89534 D0Y8UF 5040063 EC50 = 0.1 nM T89534 D0Y9BO 135461982 IC50 = 93 nM T89534 D0YH4T 10062042 IC50 = 35 nM T89534 D0YW4C 135494488 IC50 = 447 nM T89534 D0Z0UC 11638264 EC50 = 7 nM T89534 D0Z9ZY 23582387 EC50 = 1543 nM T89534 D0ZT4U 10214633 IC50 = 77 nM T45287 CK8VJ3 5311145 Ki > 600000 nM T45287 CT3L5Q 14542146 Ki = 1100000 nM T45287 CP4OT8 14542149 Ki = 57000 nM T45287 CE1P6J 15719279 Ki = 1000 nM T45287 CD28WR 15719282 Ki = 1900 nM T45287 CYR87Z 15719283 Ki > 15000 nM T45287 CS75VD 44360285 Ki = 5400 nM T45287 D0A7GO 44309732 Ki = 510 nM T12075 D03EDQ 24776445 IC50 = 15 nM T12075 C5VS0H 10098 IC50 = 500 nM T12075 CLH27B 10392802 IC50 = 100 nM T12075 C2H5XZ 25109985 IC50 > 25000 nM T12075 CXUP71 44565609 IC50 < 100 nM T12075 CTH6Y9 44565610 IC50 < 100 nM T12075 D05UKJ 442972 IC50 = 600 nM T16156 D00PEH 135449332 EC50 = 38 nM T16156 C6BF9U 2530 EC50 = 3000 nM T16156 C9Z3SR 17341 EC50 = 200 nM T16156 C6WXE2 19098 EC50 = 70 nM T16156 C74KLR 65235 EC50 = 2000 nM T16156 CUW92J 66531 EC50 = 3400 nM T16156 CO3I9C 77330 EC50 = 10000 nM T16156 CG07HK 777985 EC50 > 10000 nM T16156 CG9I1U 2737696 EC50 = 6800 nM T16156 CGON65 9824663 EC50 = 28 nM T16156 CA80GW 10364313 EC50 = 4500 nM T16156 CTV7Q4 11503128 EC50 = 244 nM T16156 C69VRE 11518094 EC50 = 640 nM T16156 CMJS98 11518228 EC50 = 60 nM T16156 CM5UR4 11525415 EC50 = 400 nM T16156 CLT9N4 11531160 EC50 = 1200 nM T16156 CEP6O1 11531618 EC50 = 400 nM T16156 CR8KX3 11532298 EC50 = 347 nM T16156 C64JCF 11532684 EC50 = 5190 nM T16156 CW8AL5 11538742 EC50 = 3000 nM T16156 CTA74D 11554024 EC50 = 1300 nM T16156 C8SOT2 11566948 EC50 > 10000 nM T16156 CRAL79 11568409 EC50 > 10000 nM T16156 CZ74NQ 11568815 EC50 = 1500 nM T16156 CY7L9V 11569630 EC50 = 54 nM T16156 C8G2NB 11576521 EC50 = 970 nM T16156 CU7O4I 11582671 EC50 = 230 nM T16156 C5RE2J 11583400 EC50 > 10000 nM T16156 CF72DG 11583454 EC50 = 410 nM T16156 CUV5S6 11584314 EC50 > 10000 nM T16156 C92QDJ 11589431 EC50 = 2260 nM T16156 CD20SM 11590685 EC50 = 120 nM T16156 C36GOV 11590686 EC50 = 320 nM T16156 C2QR4J 11596674 EC50 = 170 nM T16156 CR3G5K 11596675 EC50 > 10000 nM T16156 CM3DK9 11597753 EC50 = 8600 nM T16156 C01TWZ 11597777 EC50 = 7900 nM T16156 CFR41Z 11604181 EC50 = 3130 nM T16156 C9T2XM 11604285 EC50 = 610 nM T16156 CF3D8H 11610831 EC50 = 2560 nM T16156 CB3GC1 11612275 EC50 = 400 nM T16156 CW48GY 11612301 EC50 = 288 nM T16156 CJZ5E7 11612508 EC50 = 100 nM T16156 CXUS50 11613064 EC50 = 43 nM T16156 CN58RH 11613221 EC50 = 23 nM T16156 CL4T5J 11618419 EC50 = 720 nM T16156 C4BM8H 11619475 EC50 = 280 nM T16156 CPL9V4 11619499 EC50 = 2200 nM T16156 CYZ1X0 11619522 EC50 = 259 nM T16156 CJ2AO1 11625649 EC50 = 9000 nM T16156 C8IO6L 11626366 EC50 = 418 nM T16156 CL43SH 11626389 EC50 = 510 nM T16156 CO82EM 11627064 EC50 = 87 nM T16156 CC2T3H 11632894 EC50 = 415 nM T16156 CZ4D5B 11632921 EC50 > 10000 nM T16156 CJ2G0S 11633585 EC50 = 490 nM T16156 C67NHZ 11633622 EC50 = 7900 nM T16156 C6NKM7 11640712 EC50 > 10000 nM T16156 CCS4O1 11641136 EC50 = 100 nM T16156 C8KCG1 11641398 EC50 = 43 nM T16156 C5C6KQ 11641872 EC50 = 130 nM T16156 C1PJ2E 11642429 EC50 = 84 nM T16156 CDTO16 11653665 EC50 = 1600 nM T16156 C6M5HE 11654808 EC50 = 84 nM T16156 C8ITQ7 11655467 EC50 = 10000 nM T16156 C3YFX2 11655509 EC50 > 10000 nM T16156 CAU74N 11661454 EC50 = 568 nM T16156 CJB6S4 11663120 EC50 > 10000 nM T16156 C51UAO 11663948 EC50 = 130 nM T16156 CS3L4A 11668280 EC50 = 6800 nM T16156 CT2HA5 11675883 EC50 = 1600 nM T16156 CG83TK 11675904 EC50 = 550 nM T16156 C38YAS 11677274 EC50 > 10000 nM T16156 C6ABR1 11682586 EC50 > 10000 nM T16156 CC15UO 11684019 EC50 > 10000 nM T16156 CE28AY 11684325 EC50 = 32 nM T16156 C87BWZ 11690013 EC50 > 10000 nM T16156 CB2M4W 11696429 EC50 = 3400 nM T16156 CFV3C9 11704251 EC50 = 1300 nM T16156 C80BSK 11704904 EC50 = 4400 nM T16156 CPV1E8 11713518 EC50 = 220 nM T16156 C9HGF7 11719192 EC50 = 2300 nM T16156 CKW50X 11719880 EC50 = 33 nM T16156 CNUQ70 11720469 EC50 = 81 nM T16156 CE8PJ0 12094052 EC50 = 57 nM T16156 CVZR61 15948975 EC50 > 10000 nM T16156 C62SRV 15949077 EC50 = 253 nM T16156 CQ5FO2 15949822 EC50 = 33 nM T16156 C5GRN9 15949825 EC50 = 129 nM T16156 C1E7GD 15949911 EC50 = 294 nM T16156 C60RDP 15950250 EC50 = 430 nM T16156 C4JO7I 15950335 EC50 = 3300 nM T16156 CA1RU5 15951514 EC50 = 117 nM T16156 CX4V2G 16046749 EC50 = 127 nM T16156 CP4NI3 16046753 EC50 = 26 nM T16156 C81EZK 16046754 EC50 = 160 nM T16156 CGI6E3 16046862 EC50 = 277 nM T16156 CKC4A0 16046967 EC50 = 21 nM T16156 C9G0VC 16047073 EC50 = 449 nM T16156 C8WO4I 16047074 EC50 = 1430 nM T16156 CPNO18 16047186 EC50 = 376 nM T16156 CSK2X5 16047524 EC50 = 473 nM T16156 CTV7W2 16047530 EC50 = 333 nM T16156 CX9NW8 16047655 EC50 = 799 nM T16156 CNIS51 16047658 EC50 = 569 nM T16156 C8P4CK 16047896 EC50 = 373 nM T16156 CBHK31 16047897 EC50 = 26 nM T16156 CSYW70 16047900 EC50 = 109 nM T16156 CZX26N 16048011 EC50 = 194 nM T16156 C8EPR3 16048012 EC50 = 67 nM T16156 CG2WC4 16048013 EC50 = 65 nM T16156 CSL3U6 16048014 EC50 = 232 nM T16156 C75PNY 16048122 EC50 = 41 nM T16156 C7K0YN 16048123 EC50 = 43 nM T16156 C72BGQ 16048126 EC50 = 35 nM T16156 CU31WD 16048128 EC50 = 148 nM T16156 CI3WG9 16048235 EC50 = 284 nM T16156 CY9D4R 16048236 EC50 = 452 nM T16156 CXI05H 16048343 EC50 = 55 nM T16156 CR3W2J 16048458 EC50 = 111 nM T16156 CCZ0Q7 16062054 EC50 = 160 nM T16156 C6RWY4 16062167 EC50 = 228 nM T16156 CK6BG1 16062168 EC50 > 1000 nM T16156 CD23WV 16062169 EC50 = 51 nM T16156 CE3JQ1 16062170 EC50 = 116 nM T16156 CPS63Z 16062171 EC50 = 1260 nM T16156 CAYV13 16062172 EC50 = 179 nM T16156 CP6KL2 16659674 EC50 = 89 nM T16156 CW0DR9 17774631 EC50 = 5200 nM T16156 CAK5C6 19089431 EC50 = 1300 nM T16156 C08DIQ 24180550 EC50 = 13 nM T16156 C6IQ8G 25032375 EC50 = 25 nM T16156 CO5XN1 40480569 EC50 = 260 nM T16156 CJDT79 42636964 EC50 = 7 nM T16156 CJ10EY 44408617 EC50 = 10000 nM T16156 C7V1KA 44442626 EC50 > 10000 nM T16156 CP95WC 44442628 EC50 = 143 nM T16156 C9TF7S 44442629 EC50 = 53 nM T16156 CNBJ26 44442630 EC50 = 35 nM T16156 CQ40MJ 44442654 EC50 > 10000 nM T16156 CY0X7M 44442655 EC50 > 10000 nM T16156 C4Y3IG 44442659 EC50 = 784 nM T16156 C4D9FO 44442689 EC50 > 10000 nM T16156 CCT9W5 44442693 EC50 = 7700 nM T16156 CVZ1S3 44442698 EC50 = 540 nM T16156 CK1PE2 44442700 EC50 > 10000 nM T16156 CHKR36 44442702 EC50 > 10000 nM T16156 C70CIV 44442703 EC50 > 10000 nM T16156 C68QRW 44442705 EC50 > 10000 nM T16156 C51SLB 44442706 EC50 > 10000 nM T16156 CQ4WN5 44442710 EC50 = 38 nM T16156 CQFB05 44442713 EC50 = 65 nM T16156 CTZJ62 44442714 EC50 = 22 nM T16156 CWR7J0 44442715 EC50 = 9 nM T16156 CJ4C7Y 44442716 EC50 = 540 nM T16156 CD09GV 44442717 EC50 = 180 nM T16156 CGFA24 44442718 EC50 = 45 nM T16156 C0PH3G 44442719 EC50 = 11 nM T16156 CZ6T7E 44442720 EC50 = 140 nM T16156 C2Q4MR 44442721 EC50 = 27 nM T16156 CPO24I 44442809 EC50 > 10000 nM T16156 C3TQA4 44442810 EC50 = 6700 nM T16156 CF14EG 44442811 EC50 > 10000 nM T16156 CZ60LF 44442812 EC50 = 1400 nM T16156 C37NVG 44442813 EC50 = 2000 nM T16156 C1ZL5H 44442814 EC50 > 10000 nM T16156 CXN73O 44442815 EC50 > 10000 nM T16156 CP06FQ 44442816 EC50 > 10000 nM T16156 CBX31J 44442819 EC50 = 30 nM T16156 C3NM5G 44442823 EC50 = 71 nM T16156 C2O9VT 44442825 EC50 = 29 nM T16156 CE5R8Z 44449842 EC50 = 100 nM T16156 C9MZL8 44449843 EC50 = 89 nM T16156 C6R0OD 44449844 EC50 = 180 nM T16156 C74GBP 44449871 EC50 = 700 nM T16156 C2QKA5 44449872 EC50 = 540 nM T16156 CC6L8E 44449898 EC50 = 32 nM T16156 CG7WH6 44449907 EC50 = 530 nM T16156 C0K1XV 44449936 EC50 = 1500 nM T16156 C1CDO7 44449937 EC50 = 520 nM T16156 CC8X6D 44564570 EC50 = 57 nM T16156 C6EUW8 44564599 EC50 = 485 nM T16156 CU80OD 44564644 EC50 = 10 nM T16156 C5SY7N 44564645 EC50 = 50 nM T16156 CN1F6H 44564646 EC50 = 56 nM T16156 C4X2NJ 44564682 EC50 = 134 nM T16156 CQU1P7 44564683 EC50 = 138 nM T16156 CM8I3Q 44564684 EC50 > 1000 nM T16156 C9A8KV 44564720 EC50 > 1000 nM T16156 C6NBO9 44565185 EC50 = 28 nM T16156 CULY65 44565186 EC50 = 34 nM T16156 CFUD59 44565187 EC50 = 43 nM T16156 CKF01L 44579072 EC50 = 119 nM T16156 CV4XD6 44579073 EC50 = 76 nM T16156 CP8Z3U 44579114 EC50 > 30000 nM T16156 CM85NF 44579437 EC50 > 30000 nM T16156 CHN8Z7 44579438 EC50 > 30000 nM T16156 CHKO27 44579439 EC50 > 30000 nM T16156 C6P2SQ 44579440 EC50 = 870 nM T16156 C64QNF 44579481 EC50 = 9200 nM T16156 CKQJ84 44579482 EC50 = 143 nM T16156 CVOY95 44579556 EC50 = 7830 nM T16156 C5PJ3U 44579557 EC50 > 30000 nM T16156 C9G2YI 44579558 EC50 = 7790 nM T16156 CO4P2K 44579559 EC50 > 30000 nM T16156 C47VTJ 44579609 EC50 > 30000 nM T16156 C90HXW 44580278 EC50 = 86 nM T16156 C3L5DU 44580319 EC50 = 37 nM T16156 CG72LE 44580320 EC50 = 111 nM T16156 CTO28M 44580357 EC50 > 30000 nM T16156 C0TO5D 46911716 EC50 = 100 nM T16156 CR1Q5B 46911717 EC50 = 66 nM T16156 CJ01SF 46911718 EC50 = 58 nM T16156 CWD12T 49797998 EC50 = 702 nM T16156 CF49UI 49798018 EC50 = 86 nM T16156 CKT0H3 49798019 EC50 = 160 nM T16156 CC2Z3L 49798020 EC50 = 130 nM T16156 C5C7YA 49798044 EC50 > 898 nM T16156 CXG75P 49798045 EC50 = 574 nM T16156 C65RAN 49798046 EC50 > 811 nM T16156 C7XLO1 49798047 EC50 = 480 nM T16156 CI61BP 49798065 EC50 = 670 nM T16156 C1DAS2 49798066 EC50 > 1000 nM T16156 C4VCJ7 49798067 EC50 = 620 nM T16156 CYNB54 49798068 EC50 = 950 nM T16156 CNOL12 49798116 EC50 > 970 nM T16156 CP0Q3V 49798117 EC50 = 220 nM T16156 CZ79HB 135404155 EC50 = 900 nM T16156 C1G9TP 135404804 EC50 = 100 nM T16156 CCM1A4 135423069 EC50 = 2000 nM T16156 C0F9MB 135423098 EC50 = 7000 nM T16156 CHY6T4 135427333 EC50 = 5000 nM T16156 C87JQI 135437190 EC50 > 30000 nM T16156 CGC7F5 135437211 EC50 = 2000 nM T16156 C15EUN 135440674 EC50 = 2000 nM T16156 C1N7BD 135442106 EC50 = 5000 nM T16156 CB0DO9 135442128 EC50 = 8000 nM T16156 C6EU1Q 135444713 EC50 = 300 nM T16156 CWT65A 135450854 EC50 = 100 nM T16156 CH8X7F 135455961 EC50 = 200 nM T16156 CEK5O3 135465658 EC50 = 2000 nM T16156 CCQJ19 135470425 EC50 = 2000 nM T16156 CK3JU6 135470453 EC50 = 200 nM T16156 C5UMA1 135471629 EC50 = 300 nM T16156 CI0CL9 135475685 EC50 = 400 nM T16156 C7VY2W 135475690 EC50 = 200 nM T16156 CJ58SX 135475701 EC50 = 10000 nM T16156 CQN6L3 135484044 EC50 = 40 nM T16156 CJP7T5 135487601 EC50 = 5000 nM T16156 CE9X3L 135487637 EC50 = 1000 nM T16156 C3MF2W 135487646 EC50 = 3000 nM T16156 CB1R4P 135487683 EC50 = 2000 nM T16156 CS30LA 135492893 EC50 = 70 nM T16156 CKBJ31 135492894 EC50 = 600 nM T16156 CT1Z5O 135496743 EC50 = 300 nM T16156 CK8V4N 135509458 EC50 = 10000 nM T16156 C42FKM 135509719 EC50 = 2000 nM T16156 CG1QI3 135509739 EC50 = 300 nM T16156 CPSJ17 135512807 EC50 = 2000 nM T16156 CDY95V 135515581 EC50 = 40 nM T16156 C2XFP3 135525133 EC50 = 700 nM T16156 CL0R2K 135525134 EC50 = 500 nM T16156 C8XZ4I 135525145 EC50 = 70 nM T16156 C70YOT 135525448 EC50 = 20 nM T16156 C28OJD 135528906 EC50 > 30000 nM T16156 CW8M5E 135536046 EC50 = 3000 nM T16156 CUOB05 135542350 EC50 = 200 nM T16156 CJ45TY 135894686 EC50 = 46 nM T16156 C19CPS 136002648 EC50 = 6 nM T16156 CB5T6K 136002649 EC50 = 3 nM T16156 C42CWF 136002650 EC50 = 64 nM T16156 C70YLC 136002651 EC50 = 35 nM T16156 CD6R1Z 136002652 EC50 = 22 nM T16156 C53DPV 136002653 EC50 = 31 nM T16156 C8MV9J 136002654 EC50 = 26 nM T16156 C20ZWC 136002655 EC50 = 42 nM T16156 C7GX1C 136094780 EC50 = 2000 nM T16156 C0D1AS 136094781 EC50 = 1000 nM T16156 CYFC51 136094782 EC50 = 1000 nM T16156 C5V7TO 136094783 EC50 = 780 nM T16156 C1LW2R 136094784 EC50 = 720 nM T16156 C5R2UN 136094785 EC50 = 1750 nM T16156 CS2HN6 136094786 EC50 = 900 nM T16156 CBZ9F7 136094787 EC50 = 1600 nM T12646 D09GOS 2812 IC50 = 1400 nM T12646 D08OOJ 73051434 IC50 = 11 nM T12646 D0F6NT 1162727 IC50 > 30000 nM T12646 C05ZPG 397069 IC50 > 100000 nM T12646 C86FWD 470278 IC50 > 100000 nM T12646 C5EY0V 672872 IC50 = 80 nM T12646 CHXJ51 697280 IC50 = 190 nM T12646 CR98CN 704363 IC50 = 230 nM T12646 C1IV9D 704494 IC50 = 290 nM T12646 C4X1BC 704553 IC50 = 300 nM T12646 CYF9E1 720920 IC50 > 30000 nM T12646 C1QRW7 768027 IC50 = 2000 nM T12646 C30HYZ 788482 IC50 = 1290 nM T12646 C34XJV 793670 EC50 = 90 nM T12646 C9M6JL 863286 IC50 > 30000 nM T12646 C1KQL0 864171 IC50 > 30000 nM T12646 C8KUR0 865869 IC50 = 9920 nM T12646 C3FX5T 865870 IC50 = 2690 nM T12646 C7MLU1 877530 IC50 > 10000 nM T12646 CHX2D5 877815 IC50 = 430 nM T12646 CA0J3M 906598 IC50 > 100000 nM T12646 CD7O0J 935549 IC50 = 4800 nM T12646 CPL20I 973124 IC50 = 1300 nM T12646 CZ32JI 2249447 IC50 = 8300 nM T12646 C5Q0HK 2975404 IC50 > 37000 nM T12646 CX3JD7 3556408 IC50 = 760 nM T12646 CEM5C8 25100438 IC50 = 360 nM T12646 C07VAB 25100440 IC50 = 670 nM T12646 CDXT96 30869108 IC50 = 990 nM T12646 C1M5SP 45019715 IC50 > 30000 nM T12646 CH2V5M 46865782 IC50 = 120 nM T12646 C9P6UC 46880290 IC50 > 20000 nM T12646 CGIA46 46880328 IC50 = 2700 nM T12646 C3VKZ8 46880369 IC50 = 180 nM T12646 CZHM28 46880414 IC50 = 91 nM T12646 CAU6O0 46880464 IC50 = 120 nM T12646 CXDK90 46880466 IC50 = 140 nM T12646 CVEC92 46880467 IC50 = 170 nM T12646 CHW21A 46880468 IC50 = 190 nM T12646 C2YWI1 46880469 IC50 = 330 nM T12646 CBQ49H 46880502 IC50 = 130 nM T12646 CA6IV3 46880503 IC50 = 230 nM T12646 CZPV27 49830258 IC50 = 110 nM T12646 C7EY1H 49852176 IC50 > 5000 nM T12646 C4VIP1 50918580 IC50 = 425 nM T12646 C9OJG1 52374396 IC50 > 30000 nM T12646 CCR7O0 54670937 IC50 > 5000 nM T12646 CM59RJ 56928016 IC50 > 5000 nM T12646 CH65ZE 57328756 IC50 = 22000 nM T12646 C1XBG6 58523937 IC50 > 5000 nM T12646 C07XGU 71520305 IC50 = 88 nM T12646 CWZ27A 71520306 IC50 = 90 nM T12646 C5WQ8Z 71520307 IC50 = 100 nM T12646 CN4O3X 71520308 IC50 = 134 nM T12646 C5OK4Z 71520309 IC50 = 150 nM T12646 C6SRU5 71520310 IC50 = 184 nM T12646 C82ATI 71520425 IC50 = 225 nM T12646 C2B9KN 71520426 IC50 = 257 nM T12646 CQ1JY3 71520427 IC50 = 443 nM T12646 CZ80NI 71520429 IC50 = 43 nM T12646 CB4JG8 71520430 IC50 = 48 nM T12646 C13YPQ 71520540 IC50 = 71 nM T12646 CO2QT1 71520541 IC50 = 41 nM T12646 CI8B7L 71520542 IC50 = 42 nM T12646 CKQL06 71520543 IC50 = 63 nM T12646 CY6PL1 71520544 IC50 = 65 nM T12646 CE4Q0T 71520634 IC50 = 112 nM T12646 CMQ68E 71520635 IC50 = 162 nM T12646 CP9UY2 71520818 IC50 > 30000 nM T12646 C7HFN3 71520819 IC50 = 960 nM T12646 CS90CX 71520820 IC50 = 720 nM T12646 CPB6S5 71520821 IC50 = 960 nM T12646 C4K1AN 71520822 IC50 = 1150 nM T12646 C45XQJ 71520919 IC50 > 30000 nM T12646 C7V2LX 71520920 IC50 = 3790 nM T12646 C0F5TW 71520926 IC50 = 172 nM T12646 CBO1H8 71520927 IC50 = 262 nM T12646 C1BSM0 71520928 IC50 = 523 nM T12646 CR42SU 71520929 IC50 = 683 nM T12646 C6I0OW 71520930 IC50 = 976 nM T12646 COYE37 71520931 IC50 = 1236 nM T12646 CEHQ96 71521025 IC50 > 30000 nM T12646 C4KCX9 71521026 IC50 > 30000 nM T12646 CEYG08 71521027 IC50 > 30000 nM T12646 CU10JB 71521028 IC50 = 2250 nM T12646 C1YF8L 71521029 IC50 = 1960 nM T12646 CIG40P 71521030 IC50 = 19430 nM T12646 C5IH4G 71521031 IC50 > 30000 nM T12646 CT4O1M 71521032 IC50 = 2031 nM T12646 CH97TQ 71521033 IC50 = 536 nM T12646 CXG73H 71521034 IC50 = 379 nM T12646 CZMO73 71521035 IC50 = 1394 nM T12646 C8F3AT 71521036 IC50 = 451 nM T12646 C9YN6X 71521037 IC50 = 908 nM T12646 C27VGT 71521131 IC50 = 1880 nM T12646 CT7IQ3 71521132 IC50 = 2060 nM T12646 C1N0IP 71521133 IC50 = 2320 nM T12646 C9EJZ4 71521134 IC50 = 16220 nM T12646 C8AR7M 71521135 IC50 > 30000 nM T12646 CG1XD3 71521136 IC50 = 19600 nM T12646 C3H7PS 71521137 IC50 > 30000 nM T12646 C6X8OQ 71521138 IC50 = 71 nM T12646 C10NRW 71521139 IC50 = 58 nM T12646 C7H1ME 71521140 IC50 = 25 nM T12646 CK6M1Y 71521141 IC50 = 54 nM T12646 CI0DC4 71521236 IC50 = 2690 nM T12646 C4R3FX 71521237 IC50 = 740 nM T12646 C3AJ2W 71521238 IC50 = 960 nM T12646 CS5E0K 71521239 IC50 = 2780 nM T12646 CVSF75 71521240 IC50 = 53 nM T12646 CIY79B 71521241 IC50 = 67 nM T12646 C0K3FZ 71521347 IC50 = 2810 nM T12646 CDR29I 71521348 IC50 > 30000 nM T12646 C4P1OI 71521349 IC50 > 30000 nM T12646 C2FU7P 71521350 IC50 > 30000 nM T12646 CSP46C 71521351 IC50 > 30000 nM T12646 C2F8TA 71521352 IC50 = 470 nM T12646 CVYJ16 71521353 IC50 > 30000 nM T12646 CR1LF6 71521458 IC50 = 1290 nM T12646 CDF30Z 71521459 IC50 = 2400 nM T12646 CU9D2H 71521460 IC50 = 7730 nM T12646 C2H9UV 71521461 IC50 = 11780 nM T12646 CG8Z3S 71521462 IC50 = 26720 nM T12646 C7CF8N 71521463 IC50 > 30000 nM T12646 CM7UB5 71521536 IC50 = 440 nM T12646 C46IZM 71521537 IC50 = 18640 nM T12646 C21MUO 71521538 IC50 = 2860 nM T12646 CS43JP 71521539 IC50 = 1940 nM T12646 CMUZ53 71521540 IC50 = 8720 nM T12646 CE1FJ6 71521541 IC50 = 11170 nM T12646 CQ0BK1 71521542 IC50 > 30000 nM T12646 CBJM79 71521620 IC50 > 30000 nM T12646 CY8RF0 71521621 IC50 = 1970 nM T12646 CV4Q5F 71521622 IC50 = 4300 nM T12646 CJ9B0Z 71521623 IC50 > 30000 nM T12646 CS84PN 71521624 IC50 = 2850 nM T12646 CX6Z8C 71521625 IC50 = 3450 nM T12646 CTK92X 71521626 IC50 = 5560 nM T12646 CPF75N 71521709 IC50 = 1277 nM T12646 CPJ3Q1 71521710 IC50 = 279 nM T12646 CP82UW 71521711 IC50 = 283 nM T12646 CXRZ18 71521712 IC50 = 379 nM T12646 C3W9KG 71521713 IC50 = 524 nM T12646 CN96LY 71521714 IC50 = 3129 nM T12646 CLD68Y 71521715 IC50 = 375 nM T12646 C5WV4I 71521791 IC50 = 140 nM T12646 C93NYA 71521792 IC50 = 168 nM T12646 CSH67K 71521793 IC50 = 604 nM T12646 C7KRB8 71521794 IC50 = 220 nM T12646 C7IU9X 71521795 IC50 = 609 nM T12646 C23LYC 71521796 IC50 = 587 nM T12646 CRO46G 71521797 IC50 = 71 nM T12646 CH1KQ4 71604308 IC50 = 760 nM T12646 CEA94U 71604309 IC50 = 1100 nM T12646 CC1V2S 71607189 IC50 = 370 nM T12646 C4TG6V 72721010 IC50 = 43 nM T12646 C2R9LK 73051132 IC50 = 445 nM T12646 C1M0KD 73051133 IC50 = 153 nM T12646 CG71JS 73051280 IC50 = 47 nM T12646 C1NQ8H 73051924 IC50 = 98 nM T12646 C7IMZ0 73052240 IC50 = 3134 nM T12646 C4HM1G 73052241 IC50 = 76 nM T12646 C4FWO9 73052243 IC50 > 5000 nM T12646 C3VLG0 73052401 IC50 = 95 nM T12646 C79HDC 73052716 IC50 = 1790 nM T12646 CEG8R1 73052718 IC50 = 192 nM T12646 CTR3G9 73052878 IC50 = 6 nM T12646 C0VA6M 73053029 IC50 = 304 nM T12646 C95DXT 82192375 IC50 > 37000 nM T12646 C46GEV 89927846 IC50 = 370 nM T12646 C9W7GE 89927907 IC50 = 3000 nM T12646 CBC03Z 89927958 IC50 = 152 nM T12646 CRX36D 89927984 IC50 = 145 nM T12646 CC36BE 89928011 IC50 = 233 nM T12646 C0XAP3 89928021 IC50 = 248 nM T12646 CMI21Z 89928023 IC50 = 68 nM T12646 CYEC61 89928082 IC50 > 5000 nM T12646 C0J7BI 89928094 IC50 = 149 nM T12646 CE81KH 89928101 IC50 = 144 nM T12646 CTGD01 89928106 IC50 = 2075 nM T12646 C6WS8V 89928107 IC50 = 632 nM T12646 CK7GM3 89928109 IC50 = 795 nM T12646 CDP70Y 89928159 IC50 = 227 nM T12646 C29ART 89928200 IC50 = 342 nM T12646 C7PH3D 89928222 IC50 = 180 nM T12646 C8AZT1 89928224 IC50 = 1068 nM T12646 CBK1W6 89941289 IC50 > 5000 nM T12646 CB8IQ2 90031714 IC50 > 5000 nM T12646 CN91SG 90032051 IC50 = 651 nM T12646 CJZS64 90032070 IC50 = 367 nM T12646 CY5TU6 90032147 IC50 = 3912 nM T12646 C9ISK1 90032171 IC50 = 215 nM T12646 CNE9B5 90032547 IC50 = 8908 nM T12646 C2XC7V 90032634 IC50 = 648 nM T12646 CBTL19 101907906 IC50 = 26300 nM T12646 CA6E9Y 101910775 IC50 = 61 nM T12646 CMY30U 101910777 IC50 = 74 nM T12646 C1A8JZ 114286471 IC50 = 70 nM T12646 CMA84J 117094775 IC50 = 907 nM T12646 CF2RD3 118322226 IC50 = 4832 nM T12646 CQBG03 118724369 IC50 = 21600 nM T12646 CD71XN 118724370 IC50 = 20500 nM T12646 CEC71H 118724371 IC50 > 37000 nM T12646 CF53BA 118724372 IC50 > 37000 nM T12646 C5RFT0 118724373 IC50 = 15400 nM T12646 CH8PF1 118724374 IC50 > 37000 nM T12646 C9C4WZ 118724375 IC50 = 2600 nM T12646 C9SLR5 118724376 IC50 = 8700 nM T12646 CYX0K4 118724377 IC50 > 37000 nM T12646 COE61I 118724378 IC50 > 37000 nM T12646 CS8YZ3 118724379 IC50 = 11400 nM T12646 C9RJV7 118724380 IC50 = 4800 nM T12646 CA3LT6 118724381 IC50 > 37000 nM T12646 CE43MW 118724382 IC50 = 2700 nM T12646 CH42TP 118724383 IC50 = 2600 nM T12646 CQFZ65 118724384 IC50 = 8400 nM T12646 CYV7T4 118724385 IC50 > 37000 nM T12646 C2SV1M 118724386 IC50 = 300 nM T12646 CYLT37 118724387 IC50 = 673 nM T12646 CA93NZ 118724388 IC50 = 141 nM T12646 CV56WG 118724389 IC50 = 700 nM T12646 C7LCP1 118724390 IC50 = 3041 nM T12646 C7XV4F 118724391 IC50 = 578 nM T12646 CD2WN1 118724392 IC50 = 552 nM T12646 C9FVI6 118724393 IC50 = 483 nM T12646 C0O3AC 118724394 IC50 = 543 nM T12646 C82IQE 118724395 IC50 = 116 nM T12646 CO9R3I 118724396 IC50 = 201 nM T12646 CRF7Z9 118724397 IC50 = 879 nM T12646 C5N1SJ 118724762 IC50 = 577 nM T12646 CG01LE 118724763 IC50 = 742 nM T12646 CA39KG 118724764 IC50 = 221 nM T12646 C1JTS3 118724765 IC50 = 921 nM T12646 CK7Y9N 118724766 IC50 = 1091 nM T12646 CCM3X6 118724767 IC50 = 2189 nM T12646 CAMZ23 118724768 IC50 = 112 nM T12646 CHZ6K1 118724769 IC50 = 60 nM T12646 C5T1RV 118724770 IC50 = 150 nM T12646 CZKE26 118724771 IC50 = 570 nM T12646 CGP36N 118724772 IC50 = 1201 nM T12646 C3YPM4 118724773 IC50 = 1667 nM T12646 C3K2BJ 118724774 IC50 = 2188 nM T12646 CYJR42 118724775 IC50 = 27 nM T12646 CF5X3Y 118724776 IC50 = 36 nM T12646 C7UZ5H 118724777 IC50 = 4313 nM T12646 CO6GN4 118724778 IC50 > 10000 nM T12646 CPK72W 118724779 IC50 = 127 nM T12646 CGO35H 118724780 IC50 = 448 nM T12646 C96YAG 118724781 IC50 = 133 nM T12646 CJ1UK5 118724782 IC50 = 264 nM T12646 C8DX9G 118724783 IC50 = 986 nM T12646 CN49SF 118724784 IC50 = 9288 nM T12646 CA78KC 118724785 IC50 = 1691 nM T12646 CL25HP 118724786 IC50 = 6939 nM T12646 CEG6T2 118724787 IC50 = 7108 nM T12646 C32LRP 118724788 IC50 = 8860 nM T12646 C43QNY 118724789 IC50 = 1679 nM T12646 CCDH40 118724790 IC50 = 474 nM T12646 CA6F9K 118724791 IC50 = 2762 nM T12646 CV5P0J 118724792 IC50 = 5645 nM T12646 CWQ61D 118724793 IC50 = 4608 nM T12646 CKM04D 118724794 IC50 = 7610 nM T12646 CTRV82 118724795 IC50 = 2181 nM T12646 C69HKQ 118724796 IC50 = 2433 nM T12646 CO9W1I 118724797 IC50 = 3473 nM T12646 CLVO02 118724798 IC50 = 5036 nM T12646 CACB18 118724799 IC50 = 5165 nM T12646 C8LJ1X 118724800 IC50 > 10000 nM T12646 CCK45Q 118724801 IC50 = 46 nM T12646 C6B1FX 118724802 IC50 = 87 nM T12646 CY50JH 118724803 IC50 = 106 nM T12646 CS8O9F 118724804 IC50 = 135 nM T12646 C4SU7T 118724805 IC50 = 149 nM T12646 CW9E3Z 118724806 IC50 = 183 nM T12646 CY6C3R 118724807 IC50 = 237 nM T12646 C6H9CJ 118724808 IC50 = 59 nM T12646 CX7FM5 118724809 IC50 = 89 nM T12646 CE54NW 118724810 IC50 = 102 nM T12646 CXJ43Z 118724811 IC50 = 106 nM T12646 CVKT57 118724812 IC50 = 222 nM T12646 CZV40N 118724813 IC50 = 246 nM T12646 C4YH3Q 118724814 IC50 = 299 nM T12646 C0F8VX 118724815 IC50 = 82 nM T12646 C6QRS2 118724816 IC50 = 109 nM T12646 C3NK9E 118724817 IC50 = 452 nM T12646 C2DSR3 118724818 IC50 = 491 nM T12646 C4UJ7V 127031857 IC50 = 50 nM T12646 CT0F5Y 127032127 IC50 = 710 nM T12646 C3VG0W 127032128 IC50 = 3800 nM T12646 CGU32Y 127032429 IC50 = 4700 nM T12646 CVXR24 127032715 IC50 = 21500 nM T12646 CRN4B7 127032716 IC50 = 240 nM T12646 CKGU65 127039986 IC50 > 5000 nM T12646 CRB4C1 127039987 IC50 > 5000 nM T12646 C2GX8Z 127039988 IC50 > 5000 nM T12646 CV81YZ 127039989 IC50 = 3860 nM T12646 C6OQ4W 127039990 IC50 > 5000 nM T12646 CB2AR3 127040617 IC50 > 5000 nM T12646 CJ4FQ3 127040618 IC50 > 5000 nM T12646 CX0P2U 127040619 IC50 > 5000 nM T12646 C82QOL 127040620 IC50 > 5000 nM T12646 CWC4M7 127040621 IC50 > 5000 nM T12646 CWA09O 127040622 IC50 > 5000 nM T12646 CQ6KV5 127041309 IC50 = 15 nM T12646 CI0X6E 127041536 IC50 > 5000 nM T12646 CQ2VO1 127041608 IC50 = 71 nM T12646 CGN9I7 127041609 IC50 = 23 nM T12646 C3TUR2 127041878 IC50 > 5000 nM T12646 CR8PG7 127041879 IC50 > 5000 nM T12646 CV92NA 129073433 IC50 = 180 nM T12646 C3IN1Q 132561319 IC50 = 7900 nM T12646 C1LN3T 132570328 IC50 = 160 nM T12646 C3H6DA 132570329 IC50 = 44 nM T12646 C6H9BZ 132570331 IC50 = 31400 nM T12646 CEZ9B2 139035043 IC50 = 7200 nM T12646 CEX63L 139298248 IC50 = 7 nM T12646 C10RBQ 140939034 IC50 = 90 nM T12646 CKW53D 140939044 IC50 = 100 nM T12646 C8CQT0 140939054 IC50 = 280 nM T12646 C7TX2S 140939070 IC50 = 190 nM T12646 COWD30 140939079 IC50 = 20 nM T12646 C4V7CI 140939088 IC50 = 2610 nM T12646 C2C9PG 140939100 IC50 = 1130 nM T12646 C6PN5R 140939111 IC50 = 200 nM T12646 C0ZH4R 140939116 IC50 = 800 nM T12646 CTJ0U5 140939119 IC50 = 19000 nM T12646 CGLY18 140939126 IC50 = 210 nM T12646 CUC3P9 140939138 IC50 = 1060 nM T12646 CW8U7Q 140939163 IC50 = 4760 nM T12646 CZ0XI5 140939170 IC50 = 1050 nM T12646 CX7F5D 140939178 IC50 = 50 nM T12646 CP7Q2G 140939185 IC50 = 330 nM T12646 C4JAX8 145988686 IC50 = 380 nM T12646 C7LGD3 154730745 Ki = 33.2 nM T12646 CDN0B5 155068296 IC50 = 82.8 nM T12646 C9YQ7I 155510447 Ki = 20.8 nM T12646 C43MSR 155510502 Ki = 28.1 nM T12646 CQV4H6 155513260 Ki = 32.8 nM T12646 C3K1VZ 155513650 IC50 = 119.7 nM T12646 CSB62H 155515179 Ki = 24.5 nM T12646 CN98ID 155517954 IC50 = 922.1 nM T12646 CD0A2C 155518618 Ki = 40.8 nM T12646 CM48LB 155522046 IC50 = 34.6 nM T12646 CR34KJ 155522981 Ki = 26.6 nM T12646 C0CA1Z 155524986 Ki = 43 nM T12646 CWTP12 155527743 Ki = 32.3 nM T12646 CZA90T 155528495 IC50 = 36.4 nM T12646 C0HU1L 155528572 IC50 = 134.9 nM T12646 CG8Z9A 155530177 Ki = 30.6 nM T12646 C69LKC 155530248 Ki = 37.3 nM T12646 CBQ3N1 155533126 IC50 = 192.6 nM T12646 C80XHD 155536273 IC50 = 387.1 nM T12646 CWZS75 155538655 IC50 = 8 nM T12646 C9KO2J 155545885 IC50 = 129.4 nM T12646 C3VHG0 155547513 Ki = 42.4 nM T12646 CYFP96 155547774 Ki = 24.1 nM T12646 CLV2Z5 155555002 Ki = 26.9 nM T12646 C42ONM 155556308 IC50 = 448.7 nM T12646 C1QNZ5 155557365 Ki = 18.6 nM T12646 CGYS98 155557471 Ki = 37.9 nM T12646 CL28DA 155561627 IC50 = 160.9 nM T12646 C2M7QB 155561797 IC50 = 447.2 nM T12646 C3FXR6 155563226 IC50 = 100.9 nM T12646 C4LU8S 155563972 IC50 = 5104.5 nM T12646 CPU5R9 155564364 IC50 = 308.1 nM T12646 CIYS74 155565460 Ki = 31.4 nM T12646 D00YNY 753704 EC50 < 1200 nM T12646 D0D8SU 71521142 IC50 = 24 nM T21507 D06RWL 58448012 IC50 = 23420 nM T21507 D08SNH 71555922 Ki = 133 nM T21507 C9UH5C 78213 Ki > 10000 nM T21507 CB3K6A 96214 IC50 > 50000 nM T21507 C4FC1N 626798 Ki > 23200 nM T21507 C2B3XF 1002968 Ki = 710 nM T21507 CVC49Q 1002969 Ki = 790 nM T21507 CY1E2S 2275152 Ki = 3810 nM T21507 CPB51H 2892713 Ki = 810 nM T21507 CF2B7X 6442405 Ki > 100000 nM T21507 C5J2VI 9803569 Ki > 2000 nM T21507 CBE76H 9889814 Ki > 2000 nM T21507 C8HD1X 10001781 Ki > 2000 nM T21507 CJ4Y6Z 10031785 IC50 = 16000 nM T21507 C6NFY0 11429153 Ki > 10000 nM T21507 CN9I5J 12020821 Ki = 830 nM T21507 CO7Z8E 12020835 Ki > 2000 nM T21507 CGN02U 15038112 Ki > 10000 nM T21507 CQ81TK 17753148 Ki = 830 nM T21507 C06GWX 20577249 Ki > 2000 nM T21507 CN7GB8 20577253 Ki > 2000 nM T21507 C1WJA3 20577258 Ki > 2000 nM T21507 C7GJ4F 20577259 Ki > 2000 nM T21507 C6R9WC 20577264 Ki = 290 nM T21507 C93VWY 20577272 Ki > 2000 nM T21507 CUK06Z 20577273 Ki > 2000 nM T21507 C5USN9 20577275 Ki > 2000 nM T21507 C2HX1C 22258075 Ki = 9 nM T21507 C5N6GX 22258086 Ki < 2 nM T21507 C7PHW4 44393579 IC50 = 14000 nM T21507 CGC3D4 44393811 IC50 = 9100 nM T21507 C61CQG 44414921 Ki > 2000 nM T21507 CM5P0D 44441313 Ki = 550 nM T21507 CV8QE2 44441314 Ki = 240 nM T21507 C0LD8G 51425874 Ki = 2170 nM T21507 C9P5KT 71556166 Ki = 1200 nM T21507 C8JOU5 71556223 Ki = 500 nM T21507 C25XGY 71556353 Ki = 120 nM T21507 CP0J5L 71556425 Ki = 86 nM T21507 CB5QR3 71556493 Ki = 100 nM T21507 CIXL34 71556883 Ki = 167 nM T21507 CZ3A7E 71556887 Ki = 4300 nM T21507 CY3HG4 130428255 Ki = 2150 nM T21507 CQR81J 130428258 Ki = 2560 nM T21507 CXD7R8 130428263 Ki > 10000 nM T21507 CBLV45 130428265 Ki = 1590 nM T21507 C02NUX 130428266 Ki = 890 nM T21507 CEF56M 130428268 Ki = 770 nM T21507 CEY1U3 130428270 Ki = 1340 nM T21507 CUSP74 130428271 Ki = 3920 nM T21507 CXWQ96 130428272 Ki = 2520 nM T21507 C87ABV 130428273 Ki = 970 nM T21507 C3VUC4 130428274 Ki = 850 nM T21507 C0K4AU 130428277 Ki = 180 nM T21507 CEP6T7 130428278 Ki > 10000 nM T21507 C05DUT 130428356 Ki = 890 nM T21507 C2TD3X 130428362 Ki = 3930 nM T21507 CWZ2Q8 130428368 Ki = 550 nM T21507 CQK8P3 130428369 Ki = 1700 nM T21507 CWSI97 130428372 Ki = 680 nM T21507 C3RA1U 130428421 Ki = 1720 nM T21507 C5HV2J 130428423 Ki > 10000 nM T21507 CG76ZH 130428460 Ki = 2420 nM T21507 CDR51N 130428465 Ki = 1570 nM T21507 CBZ9F6 130428466 Ki = 1580 nM T21507 C2S9UG 145981133 Ki = 200 nM T21507 CIFQ89 145981736 Ki > 10000 nM T21507 CJ3Z6S 145982950 Ki > 10000 nM T21507 CCT63W 145983422 Ki > 10000 nM T21507 C4EF0P 145984614 Ki > 10000 nM T21507 C13NOG 145987340 Ki > 10000 nM T21507 CS2B1U 145988533 Ki > 10000 nM T21507 C1OAQ5 145989925 Ki = 2760 nM T21507 CQVR83 145991287 Ki > 10000 nM T21507 CN5MT9 145992116 Ki > 10000 nM T21507 C4SMU2 145992931 Ki > 10000 nM T21507 C4FO6M 145993680 Ki = 800 nM T21507 CVA17H 145994099 Ki = 1230 nM T21507 CR4SP9 155510891 IC50 = 20860 nM T21507 CW7Y8D 155511415 IC50 = 17130 nM T21507 CC7RL2 155517237 IC50 = 17740 nM T21507 C0W7OZ 155517587 IC50 = 4850 nM T21507 CR65JX 155520458 IC50 = 3630 nM T21507 C8PM9B 155524334 IC50 = 2760 nM T21507 C2ZVO6 155525963 IC50 = 3300 nM T21507 CS7IZ8 155526071 IC50 = 4170 nM T21507 C4KX9C 155528528 IC50 = 4610 nM T21507 CAT83B 155528650 IC50 = 15770 nM T21507 C7SEQ6 155530621 IC50 = 4190 nM T21507 CA90NS 155532366 IC50 = 8320 nM T21507 C1I3BM 155535681 IC50 = 7660 nM T21507 C3CDA5 155539479 IC50 = 10080 nM T21507 C9BD0X 155546393 IC50 = 10000 nM T21507 CV3TE6 155549399 IC50 = 30940 nM T21507 C84GMX 155554918 IC50 = 4480 nM T21507 C7ITE5 155555180 IC50 = 14630 nM T21507 C1SCP4 155555555 IC50 = 23420 nM T21507 C8RX9K 155556798 IC50 = 15960 nM T21507 C8TO2H 155559803 IC50 = 17180 nM T21507 CTL1V7 155568705 IC50 = 8120 nM T21507 CW01DA 44441441 Ki = 2 nM T21507 D00ORM 28971834 IC50 = 3000 nM T21507 D02TVS 985 Ki = 802 nM T21507 D05JAH 448769 IC50 = 6700 nM T21507 D06BBB 16122583 Ki = 350 nM T21507 D07OKT 219301 IC50 = 30000 nM T21507 D08KLL 10126984 Ki = 3 nM T21507 D0A4EA 445639 Ki = 248 nM T21507 D0B9SJ 5714537 Ki = 3400 nM T21507 D0C1DG 44393734 IC50 = 17000 nM T21507 D0WF7I 16046219 Ki = 33 nM T70792 CV03DH 51351132 IC50 = 19000 nM T70792 CH3KJ7 53317545 IC50 = 9000 nM T70792 C6URB3 53317546 IC50 = 1000 nM T70792 CYZ94I 53318830 IC50 = 100000 nM T70792 CIS49C 53321455 IC50 = 1000 nM T70792 CB0HN3 53321456 IC50 = 1000 nM T70792 CAG5V4 53321626 IC50 = 2 nM T70792 CYA84S 53322776 IC50 = 6000 nM T70792 CZ9V1F 53322777 IC50 = 1000 nM T70792 CYZ13D 53322778 IC50 = 1000 nM T70792 CF0X3D 53325416 IC50 = 100000 nM T70792 C2HX3C 53325417 IC50 = 4 nM T70792 C5PV9R 53326673 IC50 = 100000 nM T70792 CQ7XR8 53325419 IC50 = 0.4 nM T31788 CL94RI 108770 IC50 = 730 nM T31788 C4V0LT 583941 IC50 = 2300 nM T31788 C7Z1CL 659294 IC50 = 250 nM T31788 CZ2B5M 3469110 IC50 = 7900 nM T31788 C94SUH 5328791 IC50 = 43500 nM T31788 C5VIL7 10018248 IC50 = 2400 nM T31788 C0OWI9 10357192 IC50 = 1900 nM T31788 C2D3KB 14296803 IC50 = 1400 nM T31788 CR4JS7 14954965 IC50 > 30000 nM T31788 CYT0O1 34177755 IC50 > 30000 nM T31788 C1OA9Q 71667689 IC50 > 30000 nM T31788 CZ45GL 72696607 IC50 = 1250 nM T31788 C39XIK 72696608 IC50 > 30000 nM T31788 CHM0Z2 72696732 IC50 > 30000 nM T31788 CU9WS8 72696733 IC50 > 30000 nM T31788 CIO58D 72696734 IC50 > 30000 nM T31788 CDTX25 72696735 IC50 = 10 nM T31788 CK40AC 73352638 IC50 > 30000 nM T88944 C0F9KJ 16214672 EC50 = 1174.9 nM T88944 CT58GK 138319674 EC50 = 82 nM T88944 CS56CE 155511404 EC50 = 4.467 nM T88944 CHV3K9 155513302 EC50 = 5.248 nM T88944 CV21RC 155519131 EC50 = 11.75 nM T88944 C9D1LO 155526100 Ki = 602.56 nM T88944 CG2WS9 155529379 EC50 > 1000 nM T88944 CM1NS8 155534581 EC50 = 800 nM T88944 CDE02V 155538336 EC50 = 4.467 nM T88944 CDB9T5 155549840 EC50 = 3.548 nM T88944 CUX9K7 155552669 EC50 = 1300 nM T88944 CXOE70 155554720 EC50 = 0.1202 nM T88944 CX5A9S 155556159 EC50 = 8709.64 nM T88944 C8H7EF 155562158 Ki = 2511.89 nM T88944 CJ08NW 155563106 EC50 = 4570.88 nM T88944 CWTQ16 155566939 Ki = 1700 nM T88944 C8DP7O 155567021 Ki = 575.44 nM T26617 D0D0ZD 441314 IC50 = 50000 nM T26617 D0HR8Z 51634 IC50 > 100000 nM T26617 D0MU9L 176077 IC50 = 50000 nM T26617 D0RE9C 501391 IC50 = 1000000 nM T26617 D0S5LT 29435 IC50 = 62000 nM T26617 CAWL97 10888248 IC50 > 1000000 nM T26617 C06FUY 11105683 IC50 = 400000 nM T26617 CC4N0X 11258014 IC50 = 200000 nM T26617 C1JBA9 11816841 IC50 > 1000000 nM T26617 CZ21NH 23622616 IC50 = 1000000 nM T26617 CQ3SX9 44820249 IC50 = 375000 nM T26617 CNL06X 44820252 IC50 > 1000000 nM T26617 C2NXA4 101882899 IC50 = 27000 nM T26617 C05DUA 101882900 IC50 = 50000 nM T26617 CH5U7F 118411068 IC50 = 45000 nM T26617 C8X6RN 118411069 IC50 = 60000 nM T26617 C16QGB 118411070 IC50 = 80000 nM T26617 CD76NI 118411071 IC50 = 50000 nM T26617 C9LGB3 118411072 IC50 = 30000 nM T26617 CAR82K 118411073 IC50 = 20000 nM T26617 CGXZ37 118411074 IC50 = 20000 nM T26617 C8G3LO 118411076 IC50 = 17000 nM T26617 CB72ZY 118411077 IC50 > 100000 nM T26617 C2CF0W 118411108 IC50 = 125000 nM T26617 CH7BA2 118411149 IC50 = 100000 nM T26617 CUYO63 118411153 IC50 = 25000 nM T26617 CC8N6I 118719919 IC50 = 20000 nM T26617 C1WON3 118720302 IC50 = 9000 nM T26617 C0ZOT7 118720303 IC50 = 35000 nM T26617 C81YUI 118720304 IC50 > 100000 nM T26617 CXI04D 118720305 IC50 = 45000 nM T26617 CG7JV9 118720306 IC50 = 60000 nM T26617 CR4S5Y 118720307 IC50 > 100000 nM T26617 CG9Q8E 118720308 IC50 = 80000 nM T26617 D0N9IX 9822159 IC50 = 35000 nM T93515 D01BYB 5957 EC50 = 30.1 nM T93515 D03TTQ 6296 IC50 = 171000 nM T93515 D06ACW 6083 EC50 = 85 nM T93515 D07QQP 10219163 EC50 = 200 nM T93515 D0H2UB 5361 EC50 = 48000 nM T93515 D0S6AE 148197 EC50 = 60 nM T93515 D0UF2N 21706 EC50 = 145 nM T93515 D0Z7FU 6133 EC50 = 5.61 nM T93515 C9K3IP 78253 IC50 = 10000 nM T93515 CS2M9I 148196 EC50 = 100 nM T93515 C6VB7R 150973 EC50 > 1000 nM T93515 CM6QD5 189010 EC50 = 2610 nM T93515 CQX4M9 265219 IC50 > 60000 nM T93515 CCJ8P0 440317 EC50 = 1720 nM T93515 CO6A2E 451388 EC50 = 480 nM T93515 CBR21W 497297 EC50 = 1400 nM T93515 C7NR6U 3081495 EC50 >= 100000 nM T93515 COT07B 3453336 IC50 > 60000 nM T93515 C6P7VU 5311303 EC50 > 100000 nM T93515 CJ7FR1 9830339 EC50 = 830 nM T93515 CRK8Q6 9853990 EC50 = 30 nM T93515 CVZX40 9875011 EC50 = 1310 nM T93515 CR4UQ9 9875516 EC50 = 140 nM T93515 C5N9QB 9916559 EC50 = 8 nM T93515 C2F7DR 10098947 EC50 = 9400 nM T93515 CM96ZK 10168108 EC50 = 10 nM T93515 C4IV8P 10169708 EC50 = 3 nM T93515 CI9K1V 10191162 EC50 = 7 nM T93515 CN3Q7U 10207117 EC50 = 5600 nM T93515 CO0L9C 10234467 EC50 = 2270 nM T93515 C7OK5W 10255482 EC50 = 6000 nM T93515 CM4K6R 10303040 EC50 = 22 nM T93515 CF08GK 10432343 EC50 = 2000 nM T93515 CMW2L8 10929115 EC50 = 8 nM T93515 C3L6KW 10994891 EC50 = 85 nM T93515 CHB3C7 11510273 Ki = 6400 nM T93515 COI83E 11525909 EC50 = 62 nM T93515 C9M1FO 11534074 EC50 = 612 nM T93515 CT74ZJ 11560464 Ki > 15000 nM T93515 CZ8C1X 11606036 EC50 = 4900 nM T93515 CUD1J5 11611428 Ki > 15000 nM T93515 CX7J8F 11636756 IC50 = 169824.37 nM T93515 C2XOC1 11993883 EC50 > 1000 nM T93515 COZ6Y2 11993885 EC50 > 100000 nM T93515 CH4XG1 11993887 EC50 > 100000 nM T93515 CZ1J9L 11993889 EC50 <= 1000 nM T93515 CQ9ZE4 11993891 EC50 = 354 nM T93515 C3NZ6K 11994005 EC50 > 1000 nM T93515 CNBZ84 11994007 EC50 > 1000 nM T93515 CN0HI1 11994009 EC50 > 1000 nM T93515 CI48FW 11994013 EC50 > 100000 nM T93515 C2MD3V 11995641 EC50 > 1000 nM T93515 CM59TJ 11995643 EC50 > 1000 nM T93515 C67WNM 13455593 EC50 = 72 nM T93515 CUD59F 13833909 EC50 = 1600 nM T93515 C2B6HY 16082731 EC50 = 810 nM T93515 C30EVL 16114624 EC50 = 6500 nM T93515 CR6W9O 16216480 EC50 = 3 nM T93515 C3ZEI4 16655024 EC50 > 100000 nM T93515 C1QCG8 23379800 EC50 = 3670 nM T93515 C7GV8K 23662455 IC50 = 10000 nM T93515 C8KY2H 23668635 IC50 = 5430 nM T93515 C67WBS 23672996 IC50 = 5810 nM T93515 CN5OC4 23673110 IC50 = 4630 nM T93515 CA08ML 23674540 IC50 = 16200 nM T93515 CK5S9W 23686655 IC50 = 24900 nM T93515 CXZ58T 24799317 EC50 = 13940 nM T93515 CMJA06 24801414 EC50 = 13940 nM T93515 C20IDU 24857827 EC50 = 80 nM T93515 CHA2I6 24868313 IC50 = 6670 nM T93515 CNLM45 44152334 IC50 = 30300 nM T93515 C5WP3I 44157464 IC50 = 3270 nM T93515 CFB06H 44219763 EC50 = 8600 nM T93515 CTF7X3 44219764 EC50 = 1000 nM T93515 C6LSQ9 44219765 EC50 = 3400 nM T93515 CVC9D3 44306835 EC50 = 91 nM T93515 C3CU9F 44415751 EC50 > 1000 nM T93515 C9HSG4 44417696 EC50 = 564 nM T93515 C69SHE 44417704 EC50 > 100000 nM T93515 CH1OS2 44420644 EC50 = 14300 nM T93515 CIMY85 44420646 EC50 = 1880 nM T93515 C28AEV 44420650 EC50 = 470 nM T93515 COZ7M1 44420652 EC50 = 1800 nM T93515 C2D1MQ 44439743 EC50 = 31 nM T93515 CFK6P3 44439744 EC50 = 35 nM T93515 CD5F3I 44439745 EC50 = 55 nM T93515 C4OAR6 44439746 EC50 = 68 nM T93515 C53QVA 44439747 EC50 = 30 nM T93515 C3G7BR 44439748 EC50 = 221 nM T93515 CCP9D8 44439749 EC50 = 17500 nM T93515 CWTL30 44439750 EC50 = 557 nM T93515 CI18OM 44439751 EC50 = 35 nM T93515 C8LDM4 44439752 EC50 = 148 nM T93515 CIMW15 44439753 EC50 = 85 nM T93515 CEGZ01 44439754 EC50 = 77 nM T93515 C50INX 44439755 EC50 = 541 nM T93515 CSA5J1 44439756 EC50 = 88 nM T93515 CW2U7Z 44439757 EC50 = 5 nM T93515 C42YBU 44439758 EC50 = 10 nM T93515 CG6BD3 44439759 EC50 = 12 nM T93515 CI75PX 44439760 EC50 = 26 nM T93515 CYV0O8 44439761 EC50 = 140 nM T93515 C0VOD8 44439763 EC50 = 650 nM T93515 C7VHT0 44439764 EC50 = 13 nM T93515 C0IBA3 44439765 EC50 = 16 nM T93515 C81BEX 44439766 EC50 = 4 nM T93515 C39EGD 44439767 EC50 = 6 nM T93515 CFO0I8 44439812 EC50 = 42 nM T93515 CKD0G1 44439814 EC50 = 700 nM T93515 CB0G2Z 44439816 EC50 = 390 nM T93515 C4WPF7 44439818 EC50 = 200 nM T93515 CEYV61 44456046 IC50 = 3930 nM T93515 CA82XJ 44456077 IC50 = 7520 nM T93515 C1DU4Z 44456078 IC50 = 24500 nM T93515 CW9Y3A 44456081 IC50 = 11500 nM T93515 CA1DV6 44456116 IC50 = 15000 nM T93515 CHF3N0 44456160 IC50 = 9260 nM T93515 CLN38C 44456165 IC50 = 7950 nM T93515 C1W8IK 44456201 IC50 = 3040 nM T93515 CL74DQ 44457247 EC50 = 68 nM T93515 C6LWM3 44457249 EC50 = 350 nM T93515 CYB0H2 44457262 EC50 = 3070 nM T93515 CIP6B7 44457274 EC50 = 14600 nM T93515 C23NHF 44457276 EC50 = 192 nM T93515 C5Y2RW 44457290 EC50 = 94 nM T93515 CD70CI 44457294 EC50 = 52 nM T93515 C3D5SF 44457338 EC50 = 5470 nM T93515 CHS72I 44457347 EC50 = 545 nM T93515 CF8ZS7 44457361 EC50 = 130 nM T93515 CD50FC 44457390 EC50 = 13540 nM T93515 CQI0O7 44457392 EC50 = 147 nM T93515 CXO09M 44457414 EC50 = 44 nM T93515 CNW1H5 44457426 EC50 = 34 nM T93515 C6Z7JE 44457427 EC50 = 100 nM T93515 CSVR68 44457429 EC50 = 98 nM T93515 CM40ZV 44457439 EC50 = 2420 nM T93515 CD5O7G 44583580 IC50 = 12100 nM T93515 C9BM5G 44583581 IC50 = 24200 nM T93515 CJSD80 44585514 EC50 = 1890 nM T93515 C84HQM 44585515 EC50 = 5860 nM T93515 C8Q2EX 44585516 EC50 = 1880 nM T93515 C0S8XM 44585517 EC50 = 3330 nM T93515 C1V5YQ 44585518 EC50 = 300 nM T93515 C9JU8Z 44585519 EC50 = 940 nM T93515 C09XZT 44585520 EC50 > 10000 nM T93515 CRS2E1 44585521 EC50 = 3540 nM T93515 CTV7A8 44585522 EC50 = 9970 nM T93515 CXP1O4 44585523 EC50 = 7770 nM T93515 CD9A6E 44585986 EC50 = 1630 nM T93515 CR0W7K 44585987 EC50 = 794 nM T93515 CUPC35 44585988 EC50 = 910 nM T93515 CW93JX 44586005 EC50 = 1740 nM T93515 C3RS8O 44586006 EC50 = 140 nM T93515 CALX92 44586007 EC50 = 1450 nM T93515 CJHP17 44586025 EC50 = 600 nM T93515 COB6E3 44586026 EC50 = 70 nM T93515 CR57TZ 44586027 EC50 = 570 nM T93515 CV1MB6 44586042 EC50 = 3950 nM T93515 C5JV6T 44586043 EC50 = 4180 nM T93515 C08CEM 44586044 EC50 = 1700 nM T93515 C3R4LJ 44586045 EC50 = 1870 nM T93515 CIA68B 44602426 EC50 > 100000 nM T93515 C8WNI6 45104417 EC50 = 3000 nM T93515 CCT5S7 45104419 EC50 = 2000 nM T93515 C12QZE 45485253 EC50 = 3600 nM T93515 CK8QW4 46225413 IC50 > 60000 nM T93515 CJFV20 46830490 EC50 > 10000 nM T93515 CS8I2W 46830491 EC50 = 170 nM T93515 C25PCZ 46830492 EC50 = 2120 nM T93515 CK1D4T 46830493 EC50 = 2280 nM T93515 C71DNH 46831072 EC50 > 10000 nM T93515 CNR37G 46831073 EC50 > 10000 nM T93515 C2Q0RG 46831384 EC50 = 280 nM T93515 CN26KT 46831386 EC50 = 3510 nM T93515 C0B9RN 46831686 EC50 = 2130 nM T93515 CS1D6Q 46831692 EC50 = 28 nM T93515 CJQ84K 46890063 EC50 = 80 nM T93515 C0X7QY 46890111 EC50 = 16 nM T93515 C5S7CK 46890114 EC50 > 10000 nM T93515 CPCQ79 51050233 IC50 > 10000 nM T93515 C3XQD5 51050235 IC50 = 10000 nM T93515 CW0N3F 52952183 EC50 = 1800 nM T93515 CK8YW6 52952280 EC50 = 523 nM T93515 CWR0B6 52952281 EC50 = 1200 nM T93515 CHC4O2 52952282 EC50 = 6200 nM T93515 CZ86FL 52952283 EC50 = 544 nM T93515 C2DZ5A 52952391 EC50 = 907 nM T93515 CA8JY6 52952392 EC50 = 604 nM T93515 C2GNH6 52952393 EC50 = 7600 nM T93515 C2IA6G 52952394 EC50 = 2900 nM T93515 C0MWH4 52952395 EC50 = 1500 nM T93515 CZO8K6 52952396 EC50 = 4800 nM T93515 C67NQB 52952397 EC50 >= 100000 nM T93515 CBL7S0 52952494 EC50 = 1300 nM T93515 CLGF37 52952495 EC50 = 9900 nM T93515 CA3CS6 52952496 EC50 > 100000 nM T93515 CVO0A1 52952497 EC50 = 826 nM T93515 C15FQS 52952603 EC50 = 1810 nM T93515 CHR9Q8 52952604 EC50 = 1200 nM T93515 C8FUJ5 53262904 EC50 = 710 nM T93515 CA1L7N 53308118 IC50 = 24300 nM T93515 C2JIO7 53308272 EC50 = 620 nM T93515 CDH9J7 53308826 EC50 = 817 nM T93515 CJZI31 53308961 EC50 = 1500 nM T93515 CAXV23 53308962 EC50 = 6600 nM T93515 CG28DK 53309102 EC50 = 840 nM T93515 C0A1PU 53309105 EC50 = 4850 nM T93515 CG9X8W 53309242 EC50 = 3330 nM T93515 CNLP93 53309244 EC50 = 770 nM T93515 CYQ90K 53309245 EC50 = 3720 nM T93515 CR3DH9 53309379 EC50 = 2770 nM T93515 C21ZMJ 53309380 EC50 = 1890 nM T93515 CGJ86N 53309381 EC50 = 490 nM T93515 C4HL7B 53309528 EC50 = 2640 nM T93515 CDN2V9 53309529 EC50 = 500 nM T93515 CI4G5S 53309530 EC50 = 620 nM T93515 C98MFN 53326684 IC50 = 30000 nM T93515 CR98BF 53350233 IC50 > 10000 nM T93515 CGV02T 54584406 EC50 = 5000 nM T93515 C48EPI 57384078 EC50 = 400 nM T93515 CE8R4D 57384079 EC50 = 700 nM T93515 CSB13A 57384080 EC50 = 500 nM T93515 CUM6P2 57394894 EC50 = 3100 nM T93515 CL8PJ4 57394895 EC50 = 1000 nM T93515 C6U4IQ 57398422 EC50 = 2100 nM T93515 CSU2C0 57400088 EC50 > 20000 nM T93515 CJK97U 57403613 EC50 = 1500 nM T93515 C8Z5FQ 60150614 IC50 > 10000 nM T93515 C4VFI2 68530100 Ki = 2700 nM T93515 CCD47U 70685173 EC50 = 4000 nM T93515 C6WP7H 70692052 EC50 = 25900 nM T93515 C5Y4ST 70694092 EC50 = 30000 nM T93515 CLWT56 70694094 EC50 = 64200 nM T93515 C2F3LX 70694098 EC50 = 24600 nM T93515 CTEL13 71459956 EC50 = 8400 nM T93515 CH0O5B 71459957 EC50 = 5600 nM T93515 CF61BN 71459959 EC50 = 9800 nM T93515 CRD4I9 71625797 Ki > 30000 nM T93515 C2VT9G 71721777 EC50 = 840 nM T93515 C8H0CE 73348762 EC50 = 1900 nM T93515 C1I6HS 73348763 EC50 = 197 nM T93515 COQJ62 73356385 EC50 = 8400 nM T93515 CAS84P 76324375 EC50 > 100000 nM T93515 CKX98W 88151531 Ki = 1548.82 nM T93515 CES8C1 90078535 IC50 > 10000 nM T93515 C3P1MQ 90656210 EC50 = 299 nM T93515 C6CEH7 90656211 EC50 = 214 nM T93515 CVOB74 90656212 EC50 = 3400 nM T93515 CL2VA3 90656213 EC50 = 190 nM T93515 C6R2QF 90656214 EC50 = 547 nM T93515 C6PS8Q 90656215 EC50 = 350 nM T93515 CE32XG 90656216 EC50 = 325 nM T93515 CX53VO 90656217 EC50 = 187 nM T93515 C4W0IB 90656218 EC50 = 457 nM T93515 C1AD7F 90656219 EC50 = 458 nM T93515 CL9XR5 90656220 EC50 = 47 nM T93515 C93EMP 90656221 EC50 = 327 nM T93515 CJ80KG 90656222 EC50 = 285 nM T93515 CPH41T 90656223 EC50 = 103 nM T93515 CBGQ40 90656224 EC50 = 168 nM T93515 CA3X6O 90656225 EC50 = 139 nM T93515 C5VWX0 90656226 EC50 = 934 nM T93515 CFCU65 90656227 EC50 = 109 nM T93515 C5FE0D 90656230 EC50 = 66 nM T93515 C4F9RY 90656231 EC50 = 389 nM T93515 C57TEN 90656232 EC50 > 10000 nM T93515 CS7WF2 90666789 EC50 = 6200 nM T93515 CE0XU1 90666790 EC50 = 2500 nM T93515 C32TOB 90666791 EC50 = 5200 nM T93515 CNV09R 90666793 EC50 = 3300 nM T93515 CSE39Z 90666794 EC50 = 3900 nM T93515 CG29WU 90666795 EC50 = 2500 nM T93515 C40LJI 90666798 EC50 = 1700 nM T93515 C58TPX 90666799 EC50 = 2900 nM T93515 C4HT6U 90666802 EC50 = 3800 nM T93515 CMO04H 121487677 EC50 = 15500 nM T93515 C1IXO5 121487678 EC50 = 489300 nM T93515 CHIG78 132574706 IC50 = 10200 nM T93515 CA5LF2 135528590 EC50 = 140 nM T93515 C6ZB1D 137632198 IC50 = 16400 nM T93515 C4GA0J 137641946 IC50 = 13100 nM T93515 C7O3US 137643396 IC50 = 8540 nM T93515 CV24ZU 137643583 Ki = 83.18 nM T93515 CUR8V1 137648798 IC50 = 6520 nM T93515 C0UZD5 145948325 EC50 > 20000 nM T93515 CS1LP5 145948330 EC50 > 20000 nM T93515 C6Q1ZX 145948331 EC50 > 20000 nM T93515 CK41NM 145962183 Ki = 144.54 nM T93515 C8A1FO 145962191 Ki = 275.42 nM T93515 CO5Q2L 145962594 Ki = 128.82 nM T93515 CQ9B7L 145962823 Ki = 398.11 nM T93515 CXI1F8 145963427 Ki = 5248.07 nM T93515 CJ7MB8 145967007 EC50 = 3100 nM T93515 C9HK1W 145967979 EC50 = 29800 nM T93515 CL9EK8 145968441 EC50 = 10250 nM T93515 CZE31S 145971828 EC50 >= 50000 nM T93515 C5TKX8 145971893 EC50 = 26340 nM T93515 CMDI01 145978391 EC50 = 109 nM T93515 C6MG8A 90656228 EC50 = 577 nM T93515 D00PQC 6176 EC50 = 37780 nM T93515 D01PSS 65070 EC50 = 1080 nM T93515 D01ZZJ 49867142 EC50 > 100000 nM T93515 D02HAL 6031 EC50 > 10000 nM T93515 D02OAJ 5311494 EC50 = 240 nM T93515 D04IWB 10174453 EC50 = 35 nM T93515 D05MXI 42611190 IC50 > 10000 nM T93515 D05NWF 6022 EC50 > 100000 nM T93515 D06DBA 23680506 EC50 = 80.4 nM T93515 D06GQY 91934096 IC50 = 10000 nM T93515 D06PIW 53262902 EC50 = 640 nM T93515 D07LYU 53262890 EC50 = 1200 nM T93515 D07MIE 8629 EC50 = 10000 nM T93515 D07MTB 11510579 Ki > 15000 nM T93515 D07QYU 4881 EC50 > 10000 nM T93515 D07TSE 16082712 EC50 > 1000 nM T93515 D08DXA 23675622 IC50 = 11000 nM T93515 D0B0ZQ 9875920 IC50 = 1570 nM T93515 D0BB0O 121990 EC50 > 100000 nM T93515 D0DZ1K 45141593 IC50 = 29900 nM T93515 D0FF6S 16038374 IC50 > 10000 nM T93515 D0GF4I 3033941 EC50 = 26 nM T93515 D0P0EP 161647 EC50 > 100000 nM T93515 D0P4GP 52952605 EC50 = 134 nM T93515 D0P7RI 9872620 EC50 = 220 nM T93515 D0Q1HE 16116566 EC50 = 8 nM T93515 D0T4WF 11994011 EC50 > 1000 nM T93515 D0U8HD 162565 EC50 = 2300 nM T93515 D0UC4G 25090818 IC50 = 9820 nM T93515 D0Z4GJ 54210200 Ki = 21.88 nM T67812 C9A4YR 11892264 IC50 = 800 nM T67812 CM2G4X 42797508 IC50 = 16000 nM T67812 CW4Q6J 46861595 IC50 = 56 nM T67812 C36SGC 57409467 IC50 = 4 nM T67812 CY08FK 71571356 IC50 = 6.3 nM T67812 CSYP08 71602371 IC50 = 316.23 nM T67812 C49QLP 71602372 IC50 = 1.585 nM T67812 CQ1CU2 71602373 IC50 = 1995.26 nM T67812 COS59J 71602374 IC50 > 100000 nM T67812 CYE3G8 71602375 IC50 > 100000 nM T67812 CR13XU 71602433 IC50 = 19.95 nM T67812 C38SOR 71602434 IC50 = 25.12 nM T67812 C6A9OU 71602503 IC50 = 63.1 nM T67812 C3ZR8K 71603028 IC50 = 398.11 nM T67812 C9G3MW 71603091 IC50 = 7943.28 nM T67812 C7D0MK 71603092 IC50 = 5011.87 nM T67812 CP97OC 71603093 IC50 = 25.12 nM T67812 CDU53W 71603094 IC50 = 1995.26 nM T67812 CAHY94 71603095 IC50 = 63.1 nM T67812 CIYC04 71603096 IC50 = 39.81 nM T67812 C3IHF5 71603097 IC50 = 3.981 nM T67812 CNPA65 71603147 IC50 = 25.12 nM T67812 CA1EK4 71603149 IC50 = 10 nM T67812 CEI6W2 71603150 IC50 = 10000 nM T67812 CID51E 71603151 IC50 = 5011.87 nM T67812 CDK81F 71603152 IC50 = 50.12 nM T67812 C6D4JR 71603153 IC50 = 79.43 nM T67812 CRM85J 71603208 IC50 = 50.12 nM T67812 CQR5X3 71603209 IC50 = 3.162 nM T67812 CQ1K6W 71603210 IC50 > 100000 nM T67812 C9D1QC 71603211 IC50 = 398.11 nM T67812 C8JKL2 71603212 IC50 = 7943.28 nM T67812 C1S9ZW 71603213 IC50 = 251.19 nM T67812 CYS41I 71655815 IC50 = 58 nM T67812 C16EOT 71660507 IC50 = 274 nM T67812 CJTR16 71766152 IC50 > 50000 nM T67812 CJAZ61 73890915 IC50 = 3.8 nM T67812 CM4S6P 78322970 IC50 = 0.64 nM T67812 CISB78 78322972 IC50 = 1.1 nM T67812 CB3OA6 86290974 IC50 = 1 nM T67812 CR1CY4 91864584 IC50 = 0.38 nM T67812 CEC50G 91884614 IC50 = 19 nM T67812 CW1GL7 91885570 IC50 = 7.8 nM T67812 C2C4OB 91885577 IC50 = 3.1 nM T67812 CJ01BC 118262906 IC50 = 1.6 nM T67812 C95OCH 118362544 IC50 = 0.2 nM T67812 C4J9DB 118916617 IC50 > 50000 nM T67812 C8EF1P 118916631 IC50 = 4770 nM T67812 C2RBF7 118918048 IC50 > 10000 nM T67812 CN3YJ2 122179026 IC50 = 2.2 nM T67812 CSBO65 122179027 IC50 = 1 nM T67812 CWH26X 122179028 IC50 = 1.2 nM T67812 CQ54LB 122179029 IC50 = 2.1 nM T67812 C95ATE 122179030 IC50 = 41 nM T67812 C93GIX 122179031 IC50 = 170 nM T67812 CE0A2J 122179032 IC50 = 3300 nM T67812 CKDU75 122179033 IC50 = 2100 nM T67812 C8AFU6 122179034 IC50 = 23 nM T67812 CMBE26 122179035 IC50 = 3.7 nM T67812 C4WFM7 122179036 IC50 = 270 nM T67812 C04WBI 122179037 IC50 = 130 nM T67812 C2AN8V 122179038 IC50 = 6.7 nM T67812 CV2L8I 122179039 IC50 = 7.3 nM T67812 C9R6JO 122179040 IC50 = 14 nM T67812 CX6N4Q 122179041 IC50 = 3.4 nM T67812 C21ESQ 122179042 IC50 = 10 nM T67812 CWG81X 122179043 IC50 = 2.2 nM T67812 C2TS3N 122179044 IC50 = 28 nM T67812 CVN10H 122179045 IC50 = 3.6 nM T67812 CFN28S 122179046 IC50 = 2.5 nM T67812 C8XHB4 122179047 IC50 = 130 nM T67812 CZO81M 122179048 IC50 = 130 nM T67812 C63EGB 122179049 IC50 = 43 nM T67812 C8HN7U 122189249 IC50 = 30000 nM T67812 CNV03S 122189255 IC50 = 19800 nM T67812 C8UX4Q 127034759 IC50 = 760 nM T67812 CTM46H 127034938 IC50 = 2280 nM T67812 C8VYP5 127034939 IC50 > 20000 nM T67812 C4OB5T 127035411 IC50 > 10000 nM T67812 CUQ1Z6 127035947 IC50 = 5000 nM T67812 CRI96L 127035948 IC50 = 7900 nM T67812 CTN0J4 127035949 IC50 = 400 nM T67812 CZV70W 127035950 IC50 = 1440 nM T67812 CJ5OX8 127035951 IC50 = 23 nM T67812 C1M5NI 127035952 IC50 = 3600 nM T67812 C8CR0E 136662676 IC50 = 2 nM T67812 CKI37Q 137241346 IC50 = 0.3 nM T67812 CA12BF 139313440 IC50 = 0.73 nM T67812 C4MQU9 145980134 IC50 > 50000 nM T67812 CYQ67D 155515335 IC50 = 7 nM T67812 C8YF4C 155564765 IC50 < 1 nM T70633 CHDJ89 53358775 IC50 = 7 nM T70633 C37KDG 53358900 IC50 = 30 nM T70633 CUX47G 71449505 IC50 = 800 nM T70633 CZO9S6 71449506 IC50 = 1000 nM T70633 CWV05P 71449508 IC50 = 19 nM T70633 CDJ72O 71449520 IC50 = 65 nM T70633 C7JI8P 71449521 IC50 = 1000 nM T70633 CX58GV 71449522 IC50 = 3000 nM T70633 C7GTQ9 71449523 IC50 = 180 nM T70633 CN9JY4 71449524 IC50 = 2000 nM T70633 C03XDV 71451308 IC50 = 22 nM T70633 CIPT21 71451309 IC50 = 41 nM T70633 C4Y3ZU 71451310 IC50 = 200 nM T70633 C84DXS 71451316 IC50 = 3000 nM T70633 C8CG2L 71451317 IC50 > 3000 nM T70633 CA1CL3 71451318 IC50 = 160 nM T70633 CZ60YF 71453121 IC50 = 16 nM T70633 CZ7FG3 71453124 IC50 = 14 nM T70633 CDI8M1 71453125 IC50 = 720 nM T70633 CU24CR 71453138 IC50 = 90 nM T70633 CW24TS 71453139 IC50 = 300 nM T70633 CVQ2X9 71454857 IC50 = 65 nM T70633 C3H8JO 71454858 IC50 = 500 nM T70633 CP3VN0 71454869 IC50 = 700 nM T70633 C6A5OQ 71454870 IC50 = 100 nM T70633 C92QUL 71454871 IC50 = 3000 nM T70633 C62WFQ 71456626 IC50 = 300 nM T70633 CTE5Y3 71456627 IC50 = 31 nM T70633 CCH6N2 71456628 IC50 = 34 nM T70633 COI7S2 71456629 IC50 = 330 nM T70633 CC4D7M 71456641 IC50 = 40 nM T70633 C3CS5U 71456642 IC50 = 170 nM T70633 C5J1RP 71456643 IC50 = 4000 nM T70633 C4V2IW 71458486 IC50 = 17 nM T70633 C1RNK2 71458496 IC50 = 270 nM T70633 CCAM91 71458497 IC50 = 200 nM T70633 CNDT06 71458498 IC50 = 1000 nM T70633 C4WF7B 71460331 IC50 = 1000 nM T70633 CAVM60 71460332 IC50 = 11 nM T70633 C8LA3S 71460333 IC50 = 16 nM T70633 C2JS8B 71462027 IC50 = 40 nM T70633 CHOC95 71462028 IC50 = 38 nM T70633 CF31PW 71462031 IC50 = 75 nM T70633 CIE04O 71462032 IC50 = 18 nM T70633 CU5Z4N 71462033 IC50 = 49 nM T70633 CG3F6A 71462034 IC50 = 210 nM T70633 D02FGK 53358901 IC50 = 35 nM T70851 D0E3TC 44259 IC50 = 11800 nM T70851 D0WX0K 71680628 IC50 = 220 nM T70851 C26TOK 46843463 IC50 = 240 nM T70851 C8OL1N 46843542 IC50 = 200 nM T70851 C4TKF7 46843622 IC50 = 230 nM T70851 CFDB64 46843625 IC50 = 200 nM T70851 CXBA39 46843699 IC50 = 1320 nM T70851 C7RLG4 46843701 IC50 = 1240 nM T70851 CN8X2Z 46843702 IC50 = 3100 nM T70851 CU1PF4 46843771 IC50 = 200 nM T70851 C8J0HF 46843836 IC50 = 11380 nM T70851 C9GNO8 46843905 IC50 = 130 nM T70851 C1F4QN 46843908 IC50 = 320 nM T70851 CY83SC 46844092 IC50 = 260 nM T70851 C4WL6E 46844147 IC50 = 190 nM T70851 C24GBF 53319075 IC50 = 310 nM T70851 C7IT5L 53320393 IC50 = 280 nM T70851 CBC01J 53321648 IC50 = 260 nM T70851 C0F2EH 53321707 IC50 = 230 nM T70851 CBCD30 53326949 IC50 = 240 nM T70851 CV63UL 67240318 IC50 > 10000 nM T70851 CGR7I8 71604307 EC50 = 4200 nM T70851 CTDC59 73347337 EC50 > 30000 nM T70851 CHB9S7 118959070 IC50 = 700 nM T70851 CV5F2D 118959076 IC50 = 8000 nM T70851 C8L1QI 118959080 IC50 = 820 nM T70851 CX9N1Q 118959089 IC50 = 600 nM T70851 CO2L3G 118959104 IC50 = 1100 nM T70851 C0YF6P 122705989 IC50 = 8 nM T70851 C18GQC 134128280 IC50 = 35 nM T70851 C5HA8K 134610596 IC50 = 600 nM T70851 CGNO81 137333966 IC50 = 270 nM T70851 C9H2MQ 137333967 IC50 = 51 nM T70851 CR6C5X 139466406 IC50 = 170 nM T70851 C4J7ZB 139466415 IC50 = 150 nM T70851 CPN1Y4 139466419 IC50 = 9740 nM T70851 CAXL12 139466422 IC50 = 920 nM T70851 CX46RB 139466427 IC50 = 760 nM T70851 CUA8P7 139466459 IC50 = 1630 nM T70851 CNS0K3 139466461 IC50 = 210 nM T70851 CW5SE6 139466463 IC50 = 7090 nM T70851 C1G3ME 139466511 IC50 = 290 nM T70851 C7Z9ME 139466558 IC50 = 10000 nM T70851 CA5F6G 139466587 IC50 = 6700 nM T70851 C01OFP 139466597 IC50 = 530 nM T70851 C6JX9S 139466607 IC50 = 350 nM T70851 CS18LQ 139466624 IC50 = 380 nM T70851 C4V8YU 139466681 IC50 = 98 nM T70851 C6HO7F 139466682 IC50 = 2750 nM T70851 C2P6KO 139466772 IC50 = 1000 nM T70851 CU32TQ 139466793 IC50 = 7640 nM T70851 C65SUZ 139466794 IC50 = 11000 nM T70851 C0GJ3P 139473345 IC50 = 150 nM T70851 CV7UQ6 139473441 IC50 = 240 nM T70851 C4TV3Y 139473480 IC50 = 710 nM T70851 CYG76E 139473501 IC50 > 20000 nM T70851 C8RWI9 139473517 IC50 = 64 nM T70851 CBO48T 139473520 IC50 = 1660 nM T70851 CSZ85X 154701643 IC50 = 11000 nM T70851 CP5RJ6 155516750 IC50 = 2000 nM T70851 CP7SU4 155517340 IC50 > 20000 nM T70851 CF5HL4 155517637 IC50 > 20000 nM T70851 C86HPW 155518524 IC50 = 90000 nM T70851 C0L4NP 155519713 IC50 > 20000 nM T70851 CU64PX 155520421 IC50 = 30000 nM T70851 CD84CH 155521534 IC50 = 3890 nM T70851 CJ6Y8X 155522691 IC50 = 4400 nM T70851 C98ACB 155526885 IC50 = 7000 nM T70851 C6TS9K 155526919 IC50 = 18000 nM T70851 CK3F2U 155529603 IC50 = 15000 nM T70851 CS2NP9 155533143 IC50 > 20000 nM T70851 CY9SA6 155534886 IC50 > 20000 nM T70851 CX7P5O 155538726 IC50 > 120000 nM T70851 CWE36U 155544099 IC50 = 5900 nM T70851 CGKW91 155560388 IC50 > 20000 nM T70851 CSD84F 155560560 IC50 > 120000 nM T70851 C7OIS2 155561898 IC50 > 20000 nM T70851 C6WYA9 155563350 IC50 = 4100 nM T70851 C50BYF 155564479 IC50 = 40000 nM T70851 C8MOL1 155564646 IC50 = 6300 nM T70851 CXLI57 155569400 IC50 > 120000 nM T70851 D0M0QQ 46843772 IC50 = 200 nM T46456 D02DGU 444795 Ki = 1.4 nM T46456 D0G3PI 449171 IC50 = 4 nM T46456 D0N0RU 82146 Ki = 8.3 nM T46456 D06QXI 9863342 EC50 = 1 nM T46456 D08JAC 5288209 Ki > 6000 nM T46456 D09DJC 9863341 EC50 = 0.08 nM T46456 D08GRF 5287705 Ki = 9.3 nM T46456 D0YO4D 3922 Ki = 12 nM T46456 CRI78W 94391 EC50 = 42000 nM T46456 CX90MS 128016 Ki = 1000 nM T46456 C1E2FR 442048 EC50 = 33000 nM T46456 CZ8WQ4 584660 EC50 = 44000 nM T46456 CXK08W 585035 EC50 > 30000 nM T46456 CZ7K5V 585049 EC50 > 30000 nM T46456 CT30JZ 585603 EC50 > 30000 nM T46456 C9JFT3 661071 EC50 > 30000 nM T46456 CMF7L1 737267 EC50 > 30000 nM T46456 C5T2PS 843045 EC50 = 17000 nM T46456 CUHQ27 997606 EC50 > 30000 nM T46456 CZO04Y 1163179 IC50 = 18000 nM T46456 C30YVK 1169819 IC50 = 17000 nM T46456 C5UJF1 1637033 EC50 = 51000 nM T46456 CG3WZ4 2063265 EC50 > 30000 nM T46456 CG9DK0 2295706 IC50 = 18100 nM T46456 C4XZ0V 2758080 EC50 > 30000 nM T46456 C51INO 2886165 IC50 = 4900 nM T46456 CI8NO1 3025917 EC50 = 1600 nM T46456 C78QSL 3025918 EC50 = 280 nM T46456 CQ40OB 3025919 EC50 = 42 nM T46456 CYA2P5 3025934 EC50 = 1600 nM T46456 C0SBR8 3025935 EC50 = 2600 nM T46456 CK6X4W 3025936 EC50 = 1900 nM T46456 CGL71X 6366726 EC50 = 33 nM T46456 CA5GS8 6438168 EC50 = 105 nM T46456 CGTB79 6440940 EC50 = 43000 nM T46456 CJHW10 6441985 IC50 = 100 nM T46456 CVIT54 6491146 EC50 = 24000 nM T46456 CZ2N9P 7023630 EC50 = 29000 nM T46456 CG4FM8 7745122 EC50 = 1100 nM T46456 CRXY80 7745146 EC50 = 1600 nM T46456 C9SX8K 7745148 EC50 = 19000 nM T46456 CBE62R 9799320 EC50 = 71 nM T46456 COP9S7 9799477 EC50 = 4 nM T46456 CW7D0R 9810431 EC50 = 246 nM T46456 CBV6Y2 9818688 EC50 = 530 nM T46456 CEK1O4 9820039 EC50 = 160 nM T46456 CQFA96 9845057 Ki = 39 nM T46456 CQ1ZH6 9847065 Ki = 45.7 nM T46456 CAE0R3 9868664 Ki = 12.4 nM T46456 CRC51S 9869157 Ki = 40.3 nM T46456 CSK5B8 9885521 EC50 > 1000 nM T46456 C5AD1H 9886137 EC50 = 4 nM T46456 C90UXQ 9889347 Ki = 13.2 nM T46456 C8MK1Y 9889522 Ki = 620 nM T46456 C2WFX1 9905729 EC50 = 2 nM T46456 C0A3UZ 9911319 Ki = 5.6 nM T46456 C9VEF0 9949645 EC50 = 1700 nM T46456 C6JLI1 9973307 EC50 = 600 nM T46456 CVM8I3 9973559 EC50 = 26200 nM T46456 CV1A3K 9974457 EC50 > 1000 nM T46456 C7VS6O 9998151 EC50 = 520 nM T46456 CM1BQ5 10003577 Ki = 10.9 nM T46456 CZP71W 10022432 EC50 = 2600 nM T46456 C8RSG9 10043365 EC50 = 370 nM T46456 CC0N1S 10043729 EC50 = 520 nM T46456 CE60FI 10065757 Ki = 6 nM T46456 C2C0GJ 10066739 EC50 = 2300 nM T46456 CFQ1Y3 10073992 Ki = 21 nM T46456 C4VU6T 10087372 EC50 = 2600 nM T46456 CXL0Y3 10089642 EC50 = 300 nM T46456 CC8R9M 10093918 Ki = 2100 nM T46456 C59GXP 10135960 EC50 = 7 nM T46456 CO4S6H 10137005 EC50 = 99 nM T46456 CQYW32 10137940 Ki = 20 nM T46456 CP96OH 10204841 Ki = 49 nM T46456 CTKY45 10206438 Ki = 20 nM T46456 C90YNI 10207221 Ki = 37 nM T46456 C1O4PN 10207439 Ki = 20 nM T46456 C0AV2Z 10226478 Ki = 334 nM T46456 C0WRE7 10273807 Ki = 12 nM T46456 C6FT2B 10294841 EC50 = 28 nM T46456 C27ZPC 10297135 Ki = 500 nM T46456 CY1J5M 10308975 Ki = 5 nM T46456 C61TSO 10314077 EC50 = 2000 nM T46456 C6C5GP 10320109 Ki = 1000 nM T46456 C2XBM9 10362613 EC50 = 2300 nM T46456 CUEF37 10362997 IC50 = 10 nM T46456 CXA0N9 10458226 Ki = 1500 nM T46456 CL31KB 10499086 EC50 = 206 nM T46456 CF87BZ 10523774 Ki = 238 nM T46456 C2TP9D 10598286 Ki = 445 nM T46456 CS96IV 10619935 EC50 = 7 nM T46456 C4TO6H 10620598 EC50 = 9 nM T46456 CE1OC7 10644298 Ki = 467 nM T46456 CH3D5N 10645862 Ki > 1000 nM T46456 CVQ6L1 10759115 EC50 = 12500 nM T46456 C8UG3F 10926235 EC50 = 6 nM T46456 CC40ME 11793226 EC50 = 34 nM T46456 C0WA5F 11793407 Ki = 4 nM T46456 C4QYX8 11962184 Ki = 10 nM T46456 C5TS1Q 13413729 EC50 = 17100 nM T46456 CJ74NB 16794302 EC50 > 30000 nM T46456 C3P6XD 19002087 EC50 = 170 nM T46456 CVA8T2 20117108 IC50 = 6000 nM T46456 CY7P2M 20707149 EC50 = 306 nM T46456 CV1C4A 22226112 EC50 > 1000 nM T46456 CA59NU 22686157 EC50 > 30000 nM T46456 C0M9JB 22688013 EC50 = 22000 nM T46456 CP2CA5 23005221 EC50 = 220 nM T46456 C15NSJ 24828803 EC50 = 25000 nM T46456 CO31MA 24828805 EC50 = 23000 nM T46456 CW51RK 24828806 EC50 = 5600 nM T46456 C9N4PO 25195030 IC50 = 4500 nM T46456 CQUB90 25195031 IC50 = 2700 nM T46456 C0A2XU 29288275 EC50 = 10000 nM T46456 CT4J7Z 41500207 IC50 = 8200 nM T46456 CPA87R 44287651 Ki = 28 nM T46456 C1K8FB 44287715 Ki = 28 nM T46456 CI83JY 44287875 Ki = 54 nM T46456 C8W6JP 44314319 Ki > 7200 nM T46456 C17LMT 44314320 Ki > 2800 nM T46456 CH8T3V 44325132 EC50 = 86 nM T46456 C1KUN0 44325759 Ki = 172 nM T46456 CLB6X7 44325767 Ki > 1000 nM T46456 CW0T6K 44353336 Ki = 5.6 nM T46456 C8K0AB 44353347 Ki = 27.8 nM T46456 C3DYE9 44353422 Ki = 2.9 nM T46456 C5DTY3 44353441 Ki = 2.8 nM T46456 C2M8TN 44353456 Ki = 23.6 nM T46456 CVKA40 44353466 Ki = 22.5 nM T46456 C8J5SA 44353480 Ki = 27.6 nM T46456 CIB15X 44353481 Ki = 7.7 nM T46456 C1AM4Y 44377164 Ki > 1000 nM T46456 C05RAC 44377446 EC50 = 11 nM T46456 CPW0M2 44377447 EC50 = 124 nM T46456 CDU3F0 44410404 Ki = 211 nM T46456 CRW3F9 44410405 Ki = 576 nM T46456 CJX92G 44410453 Ki = 100 nM T46456 C1YKC7 44410518 Ki = 202 nM T46456 CI64YQ 44410534 Ki = 299 nM T46456 CCS4X0 44410540 Ki = 131 nM T46456 CQVY89 44410541 Ki = 35 nM T46456 CLR9U4 44410562 EC50 = 35 nM T46456 CXI98E 44410565 Ki = 31 nM T46456 C0ZIF2 44410568 Ki = 121 nM T46456 CW4YU7 44410575 Ki = 38 nM T46456 CV0TB9 44410576 Ki = 207 nM T46456 C9L6TA 44410610 EC50 = 100 nM T46456 CKY50J 44410620 Ki = 99 nM T46456 CO2AF5 44410623 Ki = 110 nM T46456 C2R7KB 44410653 Ki = 309 nM T46456 C2QW1R 44410654 EC50 = 128 nM T46456 CEA20Z 44571531 IC50 > 10000 nM T46456 CG02HN 44571532 IC50 > 10000 nM T46456 CDZ84V 44571568 IC50 = 3800 nM T46456 CF21WB 44571569 IC50 = 6600 nM T46456 CA9FT0 44571643 IC50 > 10000 nM T46456 CIO69D 59853119 EC50 = 11600 nM T46456 CNR48W 62216411 EC50 > 30000 nM T46456 C9S5EN 64222254 EC50 > 30000 nM T46456 CCX30R 71717207 Ki > 6000 nM T46456 CVW1H0 73350281 Ki = 29 nM T46456 C3PI7Z 82483008 EC50 = 24800 nM T46456 C2WG9L 138393074 EC50 = 3400 nM T46456 C2OJ9E 141259219 EC50 = 14100 nM T46456 C7N6KH 145950441 EC50 = 27200 nM T46456 CRTB69 145952096 EC50 = 2500 nM T46456 CLND09 145957286 EC50 = 50000 nM T46456 CO5LP2 145959006 EC50 = 14000 nM T46456 CM8T6X 145982686 EC50 = 17000 nM T46456 C1QZ7W 145986715 IC50 = 1800 nM T46456 C7X3AL 153763221 EC50 = 16000 nM T46456 CUNF95 155513665 EC50 = 36200 nM T46456 C3Z6VL 155514089 EC50 = 26000 nM T46456 CGO6X4 155515480 EC50 = 11000 nM T46456 CWR01U 155517898 EC50 > 30000 nM T46456 C7DN5A 155520617 EC50 > 30000 nM T46456 C95KYP 155526365 EC50 = 6400 nM T46456 C2QTX3 155530866 EC50 = 5000 nM T46456 C4JD0I 155531001 EC50 = 30000 nM T46456 CE7I8Q 155534885 EC50 = 52000 nM T46456 CE7OD6 155538138 EC50 = 1000 nM T46456 C1TMV9 155539075 EC50 = 4200 nM T46456 CEM97Q 155539095 EC50 = 21000 nM T46456 C3R9YL 155539254 EC50 = 74000 nM T46456 C7E9KD 155539294 EC50 = 4000 nM T46456 CP3I4H 155541634 EC50 = 4100 nM T46456 C2QGR5 155549327 EC50 = 21000 nM T46456 CIO4S2 155557691 EC50 = 360 nM T46456 CM52UW 155560868 EC50 = 3200 nM T46456 CG3D8J 155564760 EC50 = 3300 nM T46456 D02YHD 11755040 IC50 = 380 nM T46456 D09XCX 5694 EC50 = 31000 nM T46456 D0G6JM 5289501 IC50 > 1000 nM T46456 D0Q9FZ 6442223 EC50 = 4 nM T73696 D0Y7VM 47936 EC50 = 47 nM T73696 CS9W8Z 730108 EC50 = 94000 nM T73696 CLCE93 1313916 EC50 = 1880 nM T73696 CB32KG 1320335 EC50 = 9400 nM T73696 C9ZL4V 1511185 EC50 = 37400 nM T73696 CN3YJ7 2806493 EC50 = 1320 nM T73696 C8SW0V 4795548 EC50 = 37400 nM T73696 CA85VD 5298634 EC50 = 2360 nM T73696 C0F9KJ 16214672 EC50 > 10000 nM T73696 CXI3V4 38269206 EC50 = 13300 nM T73696 CY76JU 56593296 EC50 = 7470 nM T73696 CGJ56T 56593299 EC50 = 5290 nM T73696 C2KL3W 56593300 EC50 = 3740 nM T73696 CZNX15 56593301 EC50 = 187000 nM T73696 CX3H5E 56593302 EC50 = 59300 nM T73696 CYK15W 56593303 EC50 = 5930 nM T73696 C9CAI0 56593305 EC50 = 67 nM T73696 C34SKZ 56593306 EC50 = 4200 nM T73696 CFEB-53 56593308 EC50 = 2650 nM T73696 C1G2CT 56593309 EC50 = 1670 nM T73696 CH2OZ8 56593311 EC50 = 1880 nM T73696 CIS6Y4 56593313 EC50 = 29700 nM T73696 C86TXG 56593314 EC50 = 188 nM T73696 CG9E3B 56593316 EC50 = 52 nM T73696 C1O8DA 56593317 EC50 = 2110 nM T73696 CFD4Y1 56593318 EC50 = 2970 nM T73696 CMBL15 56593319 EC50 = 5290 nM T73696 C1WNF9 56593320 EC50 = 747 nM T73696 CZB38E 56593321 EC50 = 9400 nM T73696 CI72XF 56593322 EC50 = 47 nM T73696 C3PBI0 56593323 EC50 = 2970 nM T73696 CC86OF 56593325 EC50 = 8380 nM T73696 CZ9C4L 56593326 EC50 = 5930 nM T73696 C2KSF8 56593329 EC50 = 334 nM T73696 CE5OR0 56593330 EC50 = 188 nM T73696 CUT1H8 56593331 EC50 = 471 nM T73696 CHLI30 56593332 EC50 = 2360 nM T73696 CDM50L 56593333 EC50 = 2650 nM T73696 CD01KT 56593334 EC50 = 1060 nM T73696 C0RX7D 56593335 EC50 = 265 nM T73696 C1MDN8 56593336 EC50 = 3340 nM T73696 CIY4C2 56593337 EC50 = 3740 nM T73696 CO12YF 56593339 EC50 = 5290 nM T73696 CT1BH9 56593340 EC50 = 1880 nM T73696 CQFS58 56593342 EC50 = 94000 nM T73696 C8DNC3 56593344 EC50 = 8380 nM T73696 CVO1I9 56593345 EC50 = 747 nM T73696 CPLD89 56593346 EC50 = 1180 nM T73696 CFE3L2 56593347 EC50 = 4710 nM T73696 CIHO83 56593350 EC50 = 2660 nM T73696 CHV3K9 155513302 EC50 > 10000 nM T73696 CX5A9S 155556159 EC50 > 10000 nM T73696 CJ08NW 155563106 EC50 > 10000 nM T73696 CKXN67 155567537 EC50 > 10000 nM T73696 D01WWO 56593349 EC50 = 94 nM T21357 D05MQK 110635 IC50 > 10000 nM T21357 D0L0ZF 5663 IC50 = 14540 nM T21357 D0NJ3V 4680 Ki = 417 nM T21357 D0Y9ZE 4197 IC50 = 280 nM T21357 D01LCC 17754438 IC50 = 5360 nM T21357 D05VBJ 71295299 IC50 > 10000 nM T21357 C9LH4S 371187 IC50 = 3100 nM T21357 CZH08Y 9802738 IC50 > 20000 nM T21357 CI5GD6 9816296 IC50 = 37 nM T21357 C2AE6K 10340179 IC50 = 0.19 nM T21357 CU98NK 11518003 IC50 = 0.33 nM T21357 C9FB1N 11532490 IC50 = 4.5 nM T21357 CO2GR1 11574595 IC50 = 10 nM T21357 C0P8DN 11596587 IC50 = 0.24 nM T21357 C3G1BO 11604203 IC50 = 3850 nM T21357 C69RXL 11655838 IC50 = 0.13 nM T21357 CR8CQ7 11669507 IC50 = 23900 nM T21357 CL6F4C 11955614 Ki = 273 nM T21357 CUK49V 11988837 Ki = 1200 nM T21357 CFIO49 11988967 Ki = 1500 nM T21357 C2D0NG 11989101 Ki = 30000 nM T21357 C65ABT 11989102 Ki = 42000 nM T21357 C1B4XD 11992634 IC50 > 2000 nM T21357 CPX16N 11993169 IC50 > 2000 nM T21357 CBX53H 12805021 IC50 = 1 nM T21357 CSX70H 15991588 Ki = 463 nM T21357 C08TUE 16102593 Ki > 100 nM T21357 C7GDQ8 16102594 Ki > 100 nM T21357 CJQA32 16102595 Ki > 100 nM T21357 CHAL10 16102596 Ki < 100 nM T21357 CX0EG2 16102597 Ki = 1820 nM T21357 C6Z7GM 16102598 Ki = 328 nM T21357 C4JVF5 16102599 Ki = 280 nM T21357 CMR3A7 16102600 Ki = 237 nM T21357 CX1B4L 16102601 Ki = 332 nM T21357 CC0DP8 16102602 Ki = 207 nM T21357 CLH34A 16102603 Ki = 685 nM T21357 CK06QM 16102604 Ki = 56 nM T21357 C4TH8R 16102605 Ki = 305 nM T21357 C6X1VB 16102606 Ki = 223 nM T21357 C04SBT 16102607 Ki = 196 nM T21357 C9IK5Y 16102620 Ki < 100 nM T21357 CL6Y7J 16102621 Ki < 100 nM T21357 CNAW90 16102622 Ki = 471 nM T21357 C1GD3A 16102623 Ki = 1890 nM T21357 CX43OI 16102624 Ki = 474 nM T21357 CA52VZ 16102625 Ki = 88 nM T21357 CH25WX 16102626 Ki = 260 nM T21357 C5V1LM 16102627 Ki = 748 nM T21357 CC21RZ 16102628 Ki = 280 nM T21357 C5SN6Y 16102629 Ki = 201 nM T21357 C3S2KA 16102630 Ki = 240 nM T21357 CXFT59 17757146 IC50 = 720 nM T21357 CW96CH 21158737 IC50 = 0.11 nM T21357 CM3E7V 23647030 IC50 = 5 nM T21357 C0MO2Z 23647031 IC50 = 8.5 nM T21357 C46WZJ 23647032 IC50 = 8.8 nM T21357 CEJY54 23647042 IC50 = 2.6 nM T21357 C2CO7U 23647044 IC50 = 0.61 nM T21357 C3A7BX 23647045 IC50 = 21 nM T21357 C2YSQ6 23647046 IC50 = 0.26 nM T21357 C4M9BC 23647047 IC50 = 4.8 nM T21357 C7P2CZ 23647048 IC50 = 0.62 nM T21357 C09BFZ 23647049 IC50 = 4.8 nM T21357 CD56GP 23647050 IC50 = 10 nM T21357 C76IBZ 23647051 IC50 = 2.5 nM T21357 CE5PL6 23647052 IC50 = 3.2 nM T21357 C0IM7N 23647053 IC50 = 0.53 nM T21357 CE9L7Y 23647054 IC50 = 1.1 nM T21357 C8QZ0R 23647055 IC50 = 5.6 nM T21357 CED1K2 23647056 IC50 = 3.1 nM T21357 CN40CL 23647057 IC50 = 30 nM T21357 CBF94I 23647058 IC50 = 6.3 nM T21357 C20VHK 24871823 IC50 = 150 nM T21357 C6EQG2 24963293 IC50 > 2000 nM T21357 C4J0YD 25196719 IC50 = 4110 nM T21357 C5Q0IN 42647289 IC50 = 2300 nM T21357 CNIE98 44143458 IC50 = 4600 nM T21357 CMFN38 44351947 IC50 = 0.3 nM T21357 C7V8YH 44351948 IC50 = 0.7 nM T21357 CXC52L 44352035 IC50 = 0.7 nM T21357 C2V4KH 44352046 IC50 = 0.068 nM T21357 CKJ01T 44352047 IC50 = 0.94 nM T21357 CIM5Z7 44352055 IC50 = 0.049 nM T21357 CK7O1X 44352067 IC50 = 5.5 nM T21357 C6PZ2V 44352121 IC50 = 0.35 nM T21357 C6OJ4R 44352133 IC50 = 0.13 nM T21357 C98UBL 44452447 Ki = 1820 nM T21357 CPOZ04 44452603 Ki = 474 nM T21357 C5QCW8 46229955 IC50 = 3510 nM T21357 CFJ6O8 46229956 IC50 = 1930 nM T21357 CX85PB 46229957 IC50 = 2800 nM T21357 CG57XW 46229958 IC50 = 1140 nM T21357 CDFM64 46229998 IC50 = 1280 nM T21357 CQEK64 46229999 IC50 = 910 nM T21357 C4D5KO 46230000 IC50 = 1730 nM T21357 CX56CQ 46230001 IC50 = 1610 nM T21357 CCV17X 46230002 IC50 = 1540 nM T21357 COS0L1 46230055 IC50 = 1200 nM T21357 CR0Y7J 46230056 IC50 = 5670 nM T21357 CN41YJ 50925469 IC50 > 50000 nM T21357 CQ3RG5 50925470 IC50 > 50000 nM T21357 CS0ZD1 53324378 IC50 = 88.4 nM T21357 CHLA42 54576311 IC50 = 1250 nM T21357 C6DEG8 54576313 IC50 = 1670 nM T21357 CJF0K2 54576315 IC50 = 2510 nM T21357 CNW81G 54576317 IC50 = 2170 nM T21357 C9WEO5 54576525 IC50 = 2520 nM T21357 CD52CA 57391118 IC50 > 2000 nM T21357 CWX3N7 59320301 IC50 = 88 nM T21357 C0EP5I 59341847 IC50 = 699 nM T21357 CHQ28A 59341978 IC50 = 420 nM T21357 C4ZEH9 68578314 IC50 = 9750 nM T21357 C2HGI7 71153408 IC50 > 10000 nM T21357 C9GR3L 71153436 IC50 > 10000 nM T21357 CQ3GD7 72704434 Ki = 3100 nM T21357 CBM61I 73293715 IC50 = 107 nM T21357 CRJ8D4 90665374 IC50 = 82700 nM T21357 CG5HV8 90668361 IC50 = 16900 nM T21357 C2HQ7I 90668362 IC50 = 4800 nM T21357 CDB74T 90668364 IC50 = 3000 nM T21357 C1JPD6 91844700 IC50 = 6600 nM T21357 C5TL8H 118725359 IC50 = 6540 nM T21357 CE49ML 118725368 IC50 = 234000 nM T21357 CG0UN9 122189478 IC50 = 16720 nM T21357 CU1IF5 122189479 IC50 = 5010 nM T21357 CFK6E7 122189480 IC50 = 3830 nM T21357 CF18RV 122189481 IC50 = 5920 nM T21357 CFX0G3 122189482 IC50 = 2340 nM T21357 COT7C8 122189483 IC50 = 4650 nM T21357 CD6AS1 122189484 IC50 = 4720 nM T21357 CLJ05T 122189485 IC50 = 7270 nM T21357 CJZ8X6 122189486 IC50 = 8540 nM T21357 CMDP54 122189487 IC50 = 10210 nM T21357 C0TXZ5 122189488 IC50 = 14490 nM T21357 CZTX23 122189489 IC50 = 16620 nM T21357 CH70PC 122189490 IC50 = 25620 nM T21357 CU2ZQ6 122189491 IC50 = 25110 nM T21357 CZW60O 122189492 IC50 = 28020 nM T21357 CS6M9C 122193679 IC50 > 100000 nM T21357 CJKO62 122193703 IC50 = 103000 nM T21357 C9W1JO 122193704 IC50 = 5680 nM T21357 C2MNX0 122193705 IC50 = 19100 nM T21357 C5EHB7 122193706 IC50 = 7760 nM T21357 C5WI6U 122193707 IC50 = 4550 nM T21357 COT0R6 122193708 IC50 = 16200 nM T21357 CJF36H 122193709 IC50 = 61900 nM T21357 C0J6MS 122193710 IC50 = 29600 nM T21357 C0XLR7 122193711 IC50 = 3480 nM T21357 CC9I0U 122193712 IC50 = 3560 nM T21357 CX30HD 122193713 IC50 = 19900 nM T21357 C6IJH8 122193928 IC50 = 5610 nM T21357 CNT17O 122193929 IC50 > 1000000 nM T21357 C6Q5UO 122193930 IC50 = 50100 nM T21357 C1SWM0 122193931 IC50 = 51800 nM T21357 C9JSX0 122193932 IC50 = 28130 nM T21357 C6GI3B 122193933 IC50 = 38300 nM T21357 C9PTW4 122193934 IC50 = 16200 nM T21357 C5FKM8 122193935 IC50 = 151000 nM T21357 COA40Z 122392175 EC50 = 6000 nM T21357 C2P1IU 134129996 IC50 > 100000 nM T21357 CLE03O 134130328 IC50 > 100000 nM T21357 CSN6J0 134130563 IC50 > 100000 nM T21357 C0A1CZ 134131162 IC50 > 100000 nM T21357 C3R8SE 135457869 IC50 > 10000 nM T21357 CTX54Z 135896326 IC50 > 10000 nM T21357 C12UMG 136059728 IC50 > 1000 nM T21357 CSOF52 141737655 IC50 > 20000 nM T21357 C7SRA2 141737657 IC50 > 20000 nM T21357 CMIY07 141737666 IC50 > 20000 nM T21357 CC61SD 141737667 IC50 > 20000 nM T21357 C14CZJ 141737668 IC50 > 20000 nM T21357 CTNG49 141737674 IC50 > 20000 nM T21357 CJ38IC 141737676 IC50 > 20000 nM T21357 C1MC5Z 141737681 IC50 > 20000 nM T21357 CTUL23 141737690 IC50 > 20000 nM T21357 CMW20N 141737696 IC50 > 20000 nM T21357 CO1C4S 141737703 IC50 > 20000 nM T21357 CX9N1P 141737704 IC50 > 20000 nM T21357 C8HEG7 141737705 IC50 > 20000 nM T21357 C1S7HV 142592633 IC50 = 950 nM T21357 CN3OC2 142592634 IC50 = 169 nM T21357 CY64NR 142592636 IC50 = 321 nM T21357 C83XNL 142592649 IC50 = 800 nM T21357 CC7HN2 145974174 IC50 > 100000 nM T21357 CK1BR0 145978345 IC50 > 100000 nM T21357 CL8CU6 155521936 IC50 > 200000 nM T21357 CT85RG 155530589 IC50 > 200000 nM T21357 D0H4UN 73211886 IC50 = 24000 nM T21357 D0J0CB 2753 IC50 = 18 nM T21357 D0R6MT 3758 IC50 = 242 nM T91480 D0N5YA 65981 IC50 = 106 nM T91480 CGXS86 44394970 IC50 = 163 nM T91480 CFW4I1 44395006 IC50 = 281 nM T05849 D0L9GG 2118 IC50 > 100000 nM T05849 D0O5TQ 9853654 Ki = 14.5 nM T05849 D0U3LS 5556 IC50 > 100000 nM T05849 D04HQT 4922 IC50 = 900000 nM T05849 D04KHY 65987 IC50 = 1223 nM T05849 D0H7FW 9870520 Ki = 0.07943 nM T05849 D0LI1C 44469321 IC50 > 30000 nM T05849 D02PSZ 9962628 IC50 = 4500 nM T05849 D03OFO 9851380 IC50 > 1000 nM T05849 D0EG1F 9914672 Ki = 2.512 nM T05849 D0F6CT 51353551 IC50 = 2.7 nM T05849 D0K5UH 44381915 IC50 = 3800 nM T05849 D0RL4M 132916 IC50 = 310 nM T05849 D0W8TS 9898185 IC50 = 0.79 nM T05849 D0W9ZY 52949124 Ki = 24.55 nM T05849 D0X4AV 5311147 Ki = 0.955 nM T05849 D0XJ0S 108187 IC50 = 0.138 nM T05849 D0Y7WL 3960 IC50 = 1900 nM T05849 C6GT2N 39760 IC50 = 70000 nM T05849 C2TP7Y 104929 IC50 = 7.1 nM T05849 CCM40W 119537 IC50 > 100000 nM T05849 CXI14V 196641 IC50 = 1700 nM T05849 C3KJ7W 367893 IC50 = 170 nM T05849 C21DYZ 444998 IC50 = 170 nM T05849 C7SZ9E 613843 IC50 = 94000 nM T05849 C7YKF2 1098327 Ki = 398.11 nM T05849 CR7Y4G 1109919 Ki < 10000 nM T05849 C7WDE4 2794055 IC50 > 100000 nM T05849 CA0XN1 3081599 IC50 = 26.92 nM T05849 C83EHQ 4259649 IC50 > 100000 nM T05849 C0NT3R 4355450 IC50 = 81 nM T05849 CPM2W0 5279119 IC50 = 25000 nM T05849 CFR37P 5279123 IC50 = 52000 nM T05849 COT78N 5279169 IC50 = 270 nM T05849 C3CT7R 5279366 IC50 = 8000 nM T05849 CESY43 5279395 IC50 > 100000 nM T05849 CAD0G8 5311205 IC50 = 26.75 nM T05849 CF74HA 6918156 IC50 = 570 nM T05849 COH3V5 6957640 IC50 = 169 nM T05849 C65UQT 7216755 IC50 > 100000 nM T05849 CB80WJ 7216757 IC50 > 100000 nM T05849 CHY46J 9800177 IC50 = 40000 nM T05849 C56MLO 9802550 IC50 = 15500 nM T05849 C50RLJ 9806412 IC50 = 0.58 nM T05849 CC62IW 9808153 Ki = 36 nM T05849 CV3N7O 9823890 IC50 = 9.7 nM T05849 C2N3GQ 9828961 IC50 = 0.1 nM T05849 C6E0TB 9832467 Ki = 19.5 nM T05849 CQC1H2 9845465 IC50 = 44 nM T05849 CJL0T9 9850043 Ki = 0.3715 nM T05849 CIT4S2 9865694 IC50 = 30000 nM T05849 CD9FL8 9866980 IC50 = 1.81 nM T05849 C3UD5S 9870046 IC50 = 490 nM T05849 C1JXZ7 9875860 IC50 = 4900 nM T05849 C9I8ZU 9887120 IC50 = 130 nM T05849 C2S0NP 9896825 IC50 = 12 nM T05849 C57IBS 9913081 Ki = 25.12 nM T05849 C59XZN 9914964 IC50 = 4200 nM T05849 CK3ZO8 9934162 IC50 = 7.9 nM T05849 CR3CH6 9939183 Ki = 3.02 nM T05849 C5N8YU 9958214 Ki = 0.2089 nM T05849 CRT68S 9960432 Ki = 10 nM T05849 C53JIG 9960703 IC50 = 0.087 nM T05849 CI17HY 9962694 IC50 = 710 nM T05849 CVSE53 9977368 IC50 = 310 nM T05849 CMNI72 9978270 IC50 = 33 nM T05849 C81THG 9978327 IC50 = 14.7 nM T05849 CX74CO 9983680 IC50 = 100 nM T05849 CM31BK 9983949 Ki = 182 nM T05849 CD1GU4 9984739 IC50 = 0.6 nM T05849 C84MPA 9985004 Ki = 89 nM T05849 CHT15W 9985099 IC50 = 24 nM T05849 C0VE7T 9985100 IC50 = 4 nM T05849 C7XG4A 9985629 Ki = 51 nM T05849 CMF36V 9988096 IC50 = 6100 nM T05849 CHU9D0 9988264 IC50 = 2500 nM T05849 C0R2CH 10000984 IC50 = 632 nM T05849 C1IWA0 10001488 IC50 = 32000 nM T05849 CSCL52 10002123 IC50 = 61 nM T05849 C7F2TU 10003805 IC50 = 2.7 nM T05849 CR5AB9 10004216 Ki = 1.549 nM T05849 CCK73H 10004579 IC50 = 3.8 nM T05849 C3CZP6 10005779 IC50 = 11 nM T05849 C0KE1N 10006936 Ki = 402 nM T05849 C8X5MK 10007047 IC50 = 1.07 nM T05849 CKTR60 10008654 IC50 > 10000 nM T05849 CK05AQ 10009450 IC50 = 0.81 nM T05849 C45TFL 10009526 IC50 = 0.66 nM T05849 C2BJF9 10009604 IC50 = 30 nM T05849 CJYM64 10010723 IC50 = 42 nM T05849 CXU95K 10010811 IC50 = 12 nM T05849 CF9J4R 10010890 IC50 = 4800 nM T05849 COF3I1 10011110 IC50 = 6100 nM T05849 CVX71Q 10025585 IC50 > 100 nM T05849 C5IM3F 10027443 IC50 = 59 nM T05849 C8EYZ0 10027864 Ki < 1000 nM T05849 CPKB84 10029145 IC50 = 5.9 nM T05849 CFB8Y6 10029582 IC50 = 3.8 nM T05849 C69RVH 10030027 IC50 = 32 nM T05849 C3GZC7 10030203 IC50 = 4.4 nM T05849 CV56TJ 10031013 IC50 = 8317.64 nM T05849 CA4Y3U 10031454 Ki = 50 nM T05849 C0VXE8 10031699 IC50 = 1100 nM T05849 CD7XO3 10032955 EC50 = 2511.89 nM T05849 C7SQA8 10032956 IC50 = 177.83 nM T05849 C3KFE2 10032998 Ki = 14 nM T05849 CLQ3J6 10033396 IC50 = 4700 nM T05849 C7JIF1 10046475 IC50 = 92 nM T05849 CEX03U 10046672 IC50 = 54 nM T05849 CG2D7F 10047172 IC50 = 35 nM T05849 C0B8ZR 10047370 IC50 = 719 nM T05849 C96CLF 10047411 IC50 = 26 nM T05849 C0PI6K 10047669 IC50 = 7.5 nM T05849 C4O5CH 10048986 IC50 = 380 nM T05849 CP2FM0 10051647 IC50 = 3.4 nM T05849 CKLP95 10052234 IC50 = 13 nM T05849 CF6W7A 10053201 IC50 = 2 nM T05849 CT9PO5 10054705 Ki = 36.8 nM T05849 C3IUY0 10055040 IC50 = 50 nM T05849 C4PTZ7 10055327 IC50 = 70 nM T05849 C90VHI 10056407 IC50 = 427 nM T05849 CQM62I 10056421 IC50 = 31 nM T05849 C3JM2N 10070677 IC50 = 23 nM T05849 C4O3XJ 10070678 IC50 = 410 nM T05849 C03PUO 10070679 IC50 = 9.8 nM T05849 CFO8L6 10071178 Ki < 10000 nM T05849 CKO1P6 10071645 IC50 = 52 nM T05849 CH5YG4 10072464 Ki = 70000 nM T05849 CC84DX 10073082 IC50 = 48 nM T05849 C52HSE 10073533 IC50 = 250 nM T05849 CJ60WB 10074702 IC50 = 1 nM T05849 C4E8UF 10075014 IC50 = 1.2 nM T05849 CJ8B4F 10075052 IC50 = 6.9 nM T05849 C20EVM 10075097 IC50 = 0.24 nM T05849 CN56CR 10075297 IC50 = 48 nM T05849 CK5Y2T 10078860 Ki = 71 nM T05849 CDF7V6 10079035 IC50 = 5700 nM T05849 C5PA6Z 10079230 IC50 = 3500 nM T05849 CQ2WL5 10079315 IC50 = 3000 nM T05849 CQZ08A 10091467 IC50 = 337 nM T05849 CM81IO 10093957 IC50 = 190 nM T05849 C8CIB0 10094138 IC50 = 1200 nM T05849 CL16DK 10098459 Ki = 1.38 nM T05849 C0AG5K 10099144 IC50 = 6.7 nM T05849 CQ3KF4 10099495 Ki = 27 nM T05849 CYUX59 10099504 Ki = 134 nM T05849 CM5IG4 10101023 Ki = 40 nM T05849 CCTF24 10102593 IC50 = 10 nM T05849 CX97LH 10156187 IC50 = 28000 nM T05849 CFX06L 10182876 IC50 > 100000 nM T05849 CWR9D2 10249484 IC50 = 1070 nM T05849 C9M4LA 10252366 IC50 = 79 nM T05849 CX3M4K 10252412 IC50 = 26 nM T05849 CLF7O4 10252890 IC50 = 2300 nM T05849 CAE50W 10253366 IC50 = 220 nM T05849 CK41MD 10253387 Ki = 986 nM T05849 C3RZ6I 10253714 IC50 = 112 nM T05849 CJKQ16 10255015 Ki = 3478 nM T05849 CO7XF0 10255357 IC50 = 10.1 nM T05849 CLK7C9 10256780 Ki = 2.399 nM T05849 C1AWS5 10257790 IC50 = 0.27 nM T05849 CUN0D2 10257865 Ki = 6.1 nM T05849 CQX6S9 10258121 Ki = 20968 nM T05849 CB9W8R 10258720 IC50 = 10000 nM T05849 C0Q9IL 10258721 IC50 = 300 nM T05849 C4K3MR 10259009 IC50 = 0.45 nM T05849 CJF3O8 10260012 IC50 = 7600 nM T05849 C2ZE9N 10260074 EC50 = 130 nM T05849 CO25VX 10260206 IC50 = 7400 nM T05849 C6QI7Z 10318742 IC50 = 52 nM T05849 CO1TI7 10319892 IC50 = 5.5 nM T05849 CCFV43 10320031 IC50 = 7600 nM T05849 CPT35Q 10323073 IC50 > 100 nM T05849 C7F4SB 10323431 IC50 = 0.11 nM T05849 CAJ8S4 10323637 IC50 = 0.56 nM T05849 C2I1AN 10323690 Ki = 87 nM T05849 CMKZ57 10324322 Ki = 87 nM T05849 C17XQR 10324540 IC50 = 130 nM T05849 CUJ4E5 10325110 Ki = 79 nM T05849 CL8N3A 10327028 Ki = 15 nM T05849 C2B0ED 10341040 IC50 = 66 nM T05849 CCET87 10341247 IC50 = 5.7 nM T05849 C9V2XN 10341724 IC50 = 300 nM T05849 C9HT1U 10344702 IC50 = 192 nM T05849 C14TKQ 10345812 IC50 = 55 nM T05849 C08XGU 10346551 IC50 = 43 nM T05849 CMS8A2 10346957 IC50 = 22 nM T05849 CPL27H 10346998 IC50 = 1.5 nM T05849 CQJ56S 10347746 IC50 = 3.8 nM T05849 C2A4RZ 10349576 IC50 = 65 nM T05849 CM1D3V 10350069 IC50 = 7079.46 nM T05849 CK24IU 10350375 IC50 = 4800 nM T05849 CYT0R5 10350551 IC50 = 5200 nM T05849 CUTG21 10361419 IC50 = 38000 nM T05849 CY58LB 10363545 IC50 = 66 nM T05849 C3NK5A 10364355 IC50 = 11000 nM T05849 C2FA0Y 10364786 IC50 = 1.25 nM T05849 CE1CW5 10367509 Ki = 407 nM T05849 CZ7Y8N 10369336 IC50 = 0.6 nM T05849 CIM4A5 10369346 IC50 = 190 nM T05849 C0INE5 10369442 IC50 = 34 nM T05849 C03GYN 10369803 IC50 = 7.6 nM T05849 CF6HJ9 10369804 IC50 = 2.2 nM T05849 CL4W0M 10369805 IC50 = 0.48 nM T05849 CL3C9V 10369806 IC50 = 35.7 nM T05849 CS2J5G 10370321 Ki = 0.6607 nM T05849 CM4JF1 10371447 IC50 = 600 nM T05849 C7BT9N 10372489 Ki > 3000 nM T05849 CD6B7H 10373077 EC50 = 501.19 nM T05849 CW0G3T 10373344 IC50 = 4600 nM T05849 C7CB4V 10373378 IC50 > 10000 nM T05849 CP18HG 10389643 IC50 = 72 nM T05849 C2AYL6 10389657 IC50 = 5 nM T05849 CY18SV 10390666 Ki = 231 nM T05849 C1DR2S 10391769 IC50 = 30.4 nM T05849 CA5B8O 10391834 IC50 = 10000 nM T05849 CER5X9 10392523 IC50 = 527 nM T05849 CD8CZ6 10392653 IC50 = 8 nM T05849 C87BXC 10392698 IC50 = 7.7 nM T05849 C36LYW 10392870 IC50 = 44 nM T05849 CU4NR7 10393441 IC50 = 10.6 nM T05849 C7LD3K 10393515 Ki = 543 nM T05849 CWP78Q 10408567 IC50 = 6 nM T05849 CP7U1G 10409534 IC50 = 3 nM T05849 CT6B8X 10409900 IC50 = 6.9 nM T05849 C1F3PC 10412837 IC50 = 9.7 nM T05849 CSX57W 10413579 IC50 = 35 nM T05849 CL2IR4 10414170 IC50 = 0.28 nM T05849 CYU58T 10415786 IC50 = 15.85 nM T05849 C17ZQH 10416974 IC50 = 1.8 nM T05849 CXG5W3 10416986 IC50 = 58 nM T05849 C4FOX6 10417255 Ki = 0.8 nM T05849 CF1UI9 10418081 IC50 = 6400 nM T05849 C58UIC 10430103 IC50 = 40 nM T05849 C1U6NG 10430432 Ki = 13000 nM T05849 CENG31 10431936 IC50 = 2.2 nM T05849 CVXU85 10432393 IC50 = 300 nM T05849 CXTC17 10435698 IC50 = 1 nM T05849 CH6SG3 10436569 IC50 = 1.4 nM T05849 C03LAF 10439234 IC50 = 30 nM T05849 CG0T8U 10439779 Ki = 51 nM T05849 C0Z2QA 10440219 Ki = 39 nM T05849 C57AXJ 10440992 IC50 = 0.24 nM T05849 C8LYU6 10452597 IC50 = 32 nM T05849 C6W1ZL 10453004 IC50 = 3000 nM T05849 CD3K0I 10453063 IC50 = 137 nM T05849 CAJS89 10454826 IC50 = 15.7 nM T05849 C1MTR3 10454890 IC50 = 2900 nM T05849 CD4OL5 10455302 IC50 = 46 nM T05849 CXRI47 10455303 IC50 = 11 nM T05849 C2OAC0 10456021 IC50 = 8 nM T05849 CZ93KU 10457639 Ki > 0.0001 nM T05849 C7I8QU 10458620 IC50 = 2.5 nM T05849 CQ9M2E 10459108 IC50 = 0.22 nM T05849 CPS06J 10459641 Ki = 115 nM T05849 C3XVW4 10460621 Ki = 184 nM T05849 C7FYZ1 10462051 IC50 = 2500 nM T05849 C9Z5QY 10462206 IC50 = 600 nM T05849 CF2BH3 10463043 IC50 = 5200 nM T05849 C4PK3A 10463229 IC50 = 4250 nM T05849 C93HEO 10474221 IC50 = 2200 nM T05849 C42TBS 10475990 IC50 = 6.5 nM T05849 CT8H3X 10476766 IC50 = 4600 nM T05849 CUAV08 10477146 IC50 = 280 nM T05849 C1WQ4F 10478703 IC50 = 0.53 nM T05849 CI6UF5 10479056 IC50 = 67 nM T05849 C2YME5 10480605 IC50 = 0.074 nM T05849 C5I3TC 10481751 IC50 = 4.3 nM T05849 CEZ27H 10481933 IC50 = 3.5 nM T05849 CSOM35 10482233 Ki = 39 nM T05849 CD2O1G 10482588 IC50 = 1.4 nM T05849 CNV5G8 10482726 IC50 = 102 nM T05849 C7H4SV 10482868 Ki = 14 nM T05849 CB1X4K 10483574 IC50 = 50.12 nM T05849 CY3T4G 10484212 IC50 = 0.68 nM T05849 CQ9B2X 10484538 IC50 = 800 nM T05849 CEG0Z2 10485603 IC50 = 4500 nM T05849 CVX91R 10485763 IC50 = 6500 nM T05849 C6QR4K 10499323 IC50 > 1000 nM T05849 CNK3G4 10505959 Ki = 0.302 nM T05849 C24XLF 10506830 Ki = 33.88 nM T05849 CVE86S 10507071 IC50 = 6025 nM T05849 C91ZVY 10507109 Ki = 25.12 nM T05849 C36HIS 10507561 IC50 = 316.23 nM T05849 CJZ1T0 10508004 Ki = 1.413 nM T05849 CY0IB6 10508430 Ki > 6000 nM T05849 C03NBD 10508568 Ki = 4372 nM T05849 C9HNA2 10509035 Ki = 0.54 nM T05849 CKY68B 10509945 EC50 = 194.98 nM T05849 CZ3VH4 10526682 IC50 > 1000 nM T05849 C1AE8J 10531224 IC50 = 281.84 nM T05849 C9SUK0 10531430 IC50 = 128.82 nM T05849 C8JIW6 10532528 Ki = 3.84 nM T05849 C4H2RZ 10532660 Ki = 317 nM T05849 CF0TL3 10552320 Ki = 1.122 nM T05849 C7S9AL 10552321 Ki = 0.6761 nM T05849 C9B8PA 10554602 Ki = 0.7586 nM T05849 C4S2YR 10555164 IC50 = 478.63 nM T05849 CJZ47Q 10555363 IC50 = 794.33 nM T05849 CRI50M 10555571 IC50 = 2398.83 nM T05849 CIN1C4 10555804 IC50 = 29512.09 nM T05849 C2US6R 10555899 Ki = 0.6761 nM T05849 C38TUF 10556071 IC50 = 3840 nM T05849 CM7LP6 10556460 IC50 = 100000 nM T05849 CIEG24 10557073 Ki = 4620 nM T05849 C72MGJ 10572033 IC50 > 1000 nM T05849 C5M6NW 10576324 Ki = 2.089 nM T05849 C4TG2J 10576729 IC50 = 1.1 nM T05849 CA2B9C 10579091 Ki = 1.122 nM T05849 CJW4G1 10579208 Ki = 28 nM T05849 C6LR2W 10580108 IC50 = 8912.51 nM T05849 CW2OD9 10580252 Ki > 3000 nM T05849 CVKJ92 10580492 Ki = 1280 nM T05849 CKYT25 10597785 IC50 > 1000 nM T05849 C6B2LG 10600764 IC50 > 1000 nM T05849 CPRE54 10603576 Ki = 2.455 nM T05849 C0IT5X 10603713 IC50 = 1698.24 nM T05849 CBRX06 10603714 IC50 = 1047.13 nM T05849 CF0QX8 10604418 Ki = 1.37 nM T05849 C12XNC 10604664 Ki = 0.5623 nM T05849 CBCI69 10605398 Ki = 4.07 nM T05849 C5DMB4 10623068 Ki = 6.166 nM T05849 CIN46V 10626579 Ki = 2.884 nM T05849 C0AV6Q 10626596 IC50 = 25.12 nM T05849 CG02LF 10627173 IC50 = 5248.07 nM T05849 CF37PR 10627187 IC50 > 1000 nM T05849 C04VWM 10628422 Ki = 3.61 nM T05849 CVFQ08 10628765 Ki = 992 nM T05849 C9F2BI 10629199 Ki = 7.31 nM T05849 CF36MK 10645976 Ki = 17000 nM T05849 C46AJS 10647112 IC50 = 12 nM T05849 CIG42K 10648445 IC50 = 7.5 nM T05849 C3V8ZY 10649303 IC50 = 54 nM T05849 CWF78P 10649606 IC50 = 31.7 nM T05849 C64GDX 10650978 Ki = 63 nM T05849 CHFX82 10651325 Ki = 2.951 nM T05849 C4ZUL1 10672231 IC50 = 15 nM T05849 CR8Q4F 10673039 IC50 = 0.3 nM T05849 CXZ4C9 10675328 IC50 = 3630.78 nM T05849 CSG2H3 10676691 Ki = 95 nM T05849 CX1AF8 10676987 IC50 = 750 nM T05849 C49LHP 10695559 IC50 = 5.7 nM T05849 CGCI75 10695854 Ki = 7.762 nM T05849 C8HME7 10696336 IC50 = 1.2 nM T05849 CJA95I 10696354 Ki = 0.955 nM T05849 COQ25N 10697363 IC50 > 1000 nM T05849 C0SPI4 10697783 Ki = 4.677 nM T05849 C84WOB 10698051 IC50 = 177.83 nM T05849 C89BME 10698109 Ki = 794.33 nM T05849 CLW34G 10698427 Ki = 0.9772 nM T05849 CWMS29 10698558 Ki = 91 nM T05849 CX8P5U 10698905 IC50 = 588.84 nM T05849 C90UHA 10699165 IC50 = 1659.59 nM T05849 C9TD7U 10699583 Ki = 2.52 nM T05849 CG1KP5 10700916 EC50 > 1000 nM T05849 CMC84B 10717652 IC50 = 41 nM T05849 CKG0Q2 10719765 IC50 = 0.28 nM T05849 CN53KG 10721792 IC50 = 2630.27 nM T05849 C3R0HF 10722103 IC50 = 11220.18 nM T05849 CA9O7Y 10722372 IC50 = 39.81 nM T05849 CI4U6L 10722460 Ki = 0.8318 nM T05849 CD9G6X 10722725 Ki = 228 nM T05849 C0V1EX 10723875 Ki = 1.81 nM T05849 CC48YZ 10724082 Ki = 7.76 nM T05849 CBC78O 10739578 IC50 > 1000 nM T05849 C1A4JT 10745516 Ki = 2.344 nM T05849 CHD26N 10746778 IC50 = 158.49 nM T05849 CF9P4Z 10746830 Ki = 23.8 nM T05849 C4HD8E 10748690 IC50 = 6500 nM T05849 C3CZ6L 10748691 IC50 = 1900 nM T05849 CDK53W 10763704 IC50 > 1000 nM T05849 C8IY3W 10764164 IC50 > 1000 nM T05849 CKU83Z 10765241 IC50 = 36 nM T05849 CNJ61Y 10767360 IC50 = 26 nM T05849 CB4R1Y 10767708 Ki = 0.7244 nM T05849 C13MYE 10768190 Ki = 0.4898 nM T05849 CQ73IB 10768308 Ki = 11.48 nM T05849 C1WSH0 10768579 Ki = 0.6026 nM T05849 CK01SD 10768658 Ki = 1.95 nM T05849 CL8CO9 10769001 Ki = 0.2951 nM T05849 C7MS8F 10769675 IC50 = 190.55 nM T05849 CG1AV5 10769748 Ki = 1.318 nM T05849 C7KR4C 10769902 IC50 = 69183.1 nM T05849 C4PFX7 10770672 Ki > 3000 nM T05849 CZ2S6K 10791546 IC50 = 22 nM T05849 C8AT0Q 10792618 Ki = 0.6761 nM T05849 CJU14P 10792724 Ki = 1.549 nM T05849 C6FG8N 10792765 Ki = 0.5754 nM T05849 CZ54CL 10793342 Ki = 1.905 nM T05849 CY0WA9 10793449 Ki = 620 nM T05849 C0D9VO 10793450 Ki = 285 nM T05849 C3U6PY 10793451 Ki = 98 nM T05849 CLI85J 10793611 Ki = 60.26 nM T05849 C4G5HX 10794311 IC50 = 3.34 nM T05849 C4D6XV 10794634 Ki = 22800 nM T05849 C3R2GY 10795619 IC50 = 1400 nM T05849 C8F5HJ 10813333 IC50 = 54 nM T05849 C8AFK1 10813597 IC50 > 1000 nM T05849 C38WTD 10814625 IC50 = 0.58 nM T05849 CZ4J6S 10815094 IC50 = 20 nM T05849 CT29EW 10815832 Ki = 0.3311 nM T05849 CV2LI6 10817241 IC50 = 2951.21 nM T05849 C6EUV3 10817243 Ki = 13.18 nM T05849 C8VBP1 10817395 IC50 = 17378.01 nM T05849 CNL17K 10817407 IC50 = 724.44 nM T05849 CPER12 10819755 EC50 > 1000 nM T05849 CEZ93H 10837729 IC50 = 1.5 nM T05849 C13LGP 10838356 IC50 = 33 nM T05849 CFX92D 10838957 Ki = 0.6457 nM T05849 CTCY74 10840039 Ki = 0.7244 nM T05849 C25UOS 10841112 IC50 = 173780.08 nM T05849 C3Y6WE 10841358 IC50 = 2511.89 nM T05849 CB0I9F 10843787 IC50 = 88 nM T05849 C51ZGM 10843788 IC50 = 6500 nM T05849 C0ODR4 11027990 IC50 > 10000 nM T05849 CT7HI5 11154873 Ki = 316.23 nM T05849 CGR9A8 11178846 Ki = 125.89 nM T05849 C2O3XT 11202178 Ki = 501.19 nM T05849 C3NCV9 11212985 Ki = 316.23 nM T05849 C8WK7R 11248998 Ki = 1000 nM T05849 C72OIE 11259485 Ki = 31.62 nM T05849 CY75OQ 11271596 Ki = 794.33 nM T05849 CVL2X8 11281656 Ki = 251.19 nM T05849 C2ZUE8 11292979 Ki = 7943.28 nM T05849 CL38VT 11293780 Ki = 158.49 nM T05849 CD4I0A 11305046 Ki = 316.23 nM T05849 CKL0X6 11316421 Ki = 630.96 nM T05849 CBNS24 11316813 Ki = 158.49 nM T05849 C9VA4Z 11352971 Ki = 31.62 nM T05849 CU75AT 11353036 Ki = 5.012 nM T05849 C93AYP 11362153 Ki = 1000 nM T05849 C3QE5S 11362975 Ki = 125.89 nM T05849 COG3H2 11363465 Ki = 31.62 nM T05849 C9DF4G 11363566 Ki = 63.1 nM T05849 CXH69E 11385416 Ki = 63.1 nM T05849 C9IX1T 11396307 Ki = 251.19 nM T05849 CRA51C 11420366 Ki = 158.49 nM T05849 COSZ16 11430523 Ki = 1000 nM T05849 CT0RI9 11431264 Ki = 1258.93 nM T05849 CXIN31 11442229 Ki = 794.33 nM T05849 C9U8VO 11453391 Ki = 39.81 nM T05849 C6AYO0 11454197 Ki = 63.1 nM T05849 CE96SJ 11464858 Ki = 79.43 nM T05849 C58JUC 11465671 Ki = 63.1 nM T05849 CF9U1W 11511721 Ki = 6.026 nM T05849 CT34FE 11512112 Ki = 288.4 nM T05849 CV02EM 11512151 Ki = 7943.28 nM T05849 C9TE6V 11527738 Ki = 1 nM T05849 CYF52S 11534407 Ki = 501.19 nM T05849 C21ELY 11534594 Ki > 10000 nM T05849 C5Z9QG 11540402 Ki = 8.913 nM T05849 CA8WL2 11541048 Ki = 501.19 nM T05849 C7QYJ1 11555166 Ki = 13.18 nM T05849 C16KZS 11556194 Ki = 158.49 nM T05849 CW14OF 11576771 Ki = 26.92 nM T05849 C8B2SH 11584582 Ki = 1584.89 nM T05849 CK4H5O 11584903 Ki = 29.51 nM T05849 CU2MO1 11591504 Ki = 5.495 nM T05849 C24OIW 11592162 Ki = 44.67 nM T05849 CN6AR3 11605814 Ki = 7.943 nM T05849 CT29GZ 11613982 Ki = 15.85 nM T05849 CO3F1P 11627917 Ki = 630.96 nM T05849 CLE1G0 11628273 Ki = 16.6 nM T05849 C4EHB7 11635377 Ki = 501.19 nM T05849 CTK13M 11642370 Ki = 9.12 nM T05849 COM97A 11656338 Ki = 15.14 nM T05849 CK1O2Z 11663308 Ki = 74.13 nM T05849 CK61JR 11663565 Ki = 6.026 nM T05849 CW79UI 11693225 Ki = 25.12 nM T05849 C2P8MQ 11699148 Ki = 2511.89 nM T05849 C42YZA 11700410 Ki = 5.012 nM T05849 CFN95V 11705988 Ki = 194.98 nM T05849 CV9M3K 11712880 Ki = 13.18 nM T05849 C37SIO 11729474 IC50 = 121 nM T05849 CHK0M4 11741582 IC50 = 860 nM T05849 C3KGC7 11742520 IC50 = 1200 nM T05849 CBSD18 11742839 IC50 = 144 nM T05849 CP90MG 11744065 IC50 = 500 nM T05849 CJH86K 11753772 IC50 = 26 nM T05849 CDBF59 11756709 IC50 = 7.2 nM T05849 C5MF8W 11757086 IC50 = 5.6 nM T05849 CAZD47 11758349 IC50 > 10000 nM T05849 CX9L4P 11764851 IC50 = 10000 nM T05849 CD2E1C 11765121 IC50 = 3.3 nM T05849 C65DTB 11765552 IC50 = 223.87 nM T05849 CSX23A 11786290 Ki = 10 nM T05849 CMZG57 11798410 IC50 > 1000 nM T05849 CV4DY9 11798691 IC50 = 0.2 nM T05849 C78NMR 11799257 Ki = 8.318 nM T05849 C18WSA 11801315 Ki = 1.259 nM T05849 C8L2NZ 11801335 IC50 = 31.62 nM T05849 CN5KD0 11801461 Ki = 791 nM T05849 C6UX4C 11801462 Ki = 330 nM T05849 CSH7X6 11801911 IC50 = 776.25 nM T05849 C3SI1A 11803482 Ki = 2.7 nM T05849 C0ZPQ6 11803697 IC50 = 1200 nM T05849 C6PS4B 11803746 IC50 = 150 nM T05849 C9G7WE 13178389 IC50 = 25 nM T05849 CP7J1A 13605417 IC50 = 5600 nM T05849 CQP20O 13809511 IC50 = 26000 nM T05849 CT20PV 13809514 IC50 > 40000 nM T05849 CTS2I7 13822910 IC50 > 100000 nM T05849 CZT86R 13822916 IC50 = 12000 nM T05849 C9A4YN 13822921 IC50 = 2400 nM T05849 CAZ7H9 13822922 IC50 = 65 nM T05849 CNQ02L 13822923 IC50 = 7 nM T05849 CXI9V4 13822924 IC50 = 3000 nM T05849 C0B5DL 13953692 IC50 = 25000 nM T05849 C1Z7NU 13953694 IC50 > 100000 nM T05849 C9H0RN 13953696 IC50 > 100000 nM T05849 C5J0RC 13953698 IC50 = 60000 nM T05849 CL9Q4C 13953709 IC50 = 4800 nM T05849 C61ORP 13953715 IC50 = 380 nM T05849 CKCI39 13953716 IC50 = 380 nM T05849 C4AEO9 14030796 IC50 = 300 nM T05849 C6RT0C 14154723 IC50 = 25000 nM T05849 CMF30H 14208192 IC50 = 4000 nM T05849 CZ05OR 14208194 IC50 = 1400 nM T05849 C9WM1D 14208197 IC50 > 100000 nM T05849 CNDY74 14208198 IC50 > 100000 nM T05849 CC28YX 14208199 IC50 = 18000 nM T05849 CS3GZ8 14208200 IC50 = 17000 nM T05849 CEZ28U 14208202 IC50 = 3900 nM T05849 CNE6M7 14208204 IC50 = 14000 nM T05849 CCRZ68 14208205 IC50 > 10000 nM T05849 C95CUY 14208206 IC50 > 10000 nM T05849 CN26QE 14208208 IC50 = 3800 nM T05849 CUWX86 14208210 IC50 = 11000 nM T05849 CO0VN7 14208211 IC50 > 40000 nM T05849 CL68OI 14208212 IC50 = 110000 nM T05849 CYI95A 14208213 IC50 = 25000 nM T05849 COSQ82 14208214 IC50 = 14000 nM T05849 CD54MZ 14208215 IC50 = 29000 nM T05849 C4DFM9 14208216 IC50 = 11000 nM T05849 CX5QY0 14208217 IC50 > 10000 nM T05849 C31PLA 14208220 IC50 = 25000 nM T05849 C9PC8E 14208221 IC50 = 2900 nM T05849 C9HAS5 14208225 IC50 = 28 nM T05849 CD5EB1 14208226 IC50 = 240 nM T05849 C1U8QJ 14208227 IC50 = 1600 nM T05849 CPON92 14208228 IC50 = 390 nM T05849 C06SBR 14208229 IC50 > 10000 nM T05849 C61QZS 14208230 IC50 = 20000 nM T05849 CH7OP3 14208231 IC50 = 15000 nM T05849 C9M2XR 14208232 IC50 = 650 nM T05849 CBU7Q1 14208233 IC50 > 10000 nM T05849 CY4SV8 14208234 IC50 = 29000 nM T05849 CJ9U4R 14208235 IC50 > 10000 nM T05849 CHZ4I8 14208236 IC50 = 6300 nM T05849 C2P6RF 14208237 IC50 = 120 nM T05849 CZV4C2 14208238 IC50 > 100000 nM T05849 CW3R9Q 14208239 IC50 > 10000 nM T05849 C6RHK0 14208240 IC50 > 10000 nM T05849 C8VAY7 14208241 IC50 = 800 nM T05849 CZFH81 14208242 IC50 = 690 nM T05849 C36GAC 14208243 IC50 = 6700 nM T05849 CA94NM 14208244 IC50 = 2900 nM T05849 CX36ZB 14208245 IC50 = 8200 nM T05849 CY74SB 14208246 IC50 = 18000 nM T05849 C1UYA8 14208247 IC50 = 8200 nM T05849 CYO09N 14208248 IC50 = 9500 nM T05849 C8ZW3F 14208249 IC50 = 5000 nM T05849 C1ZE2W 14208250 IC50 = 30000 nM T05849 CGP9U0 14208251 IC50 = 7500 nM T05849 CDZ4I9 14208252 IC50 = 130000 nM T05849 C2IY4X 14208253 IC50 = 19000 nM T05849 CU8JZ3 14208254 IC50 = 5400 nM T05849 CRO59W 14208255 IC50 > 100000 nM T05849 CNH0M3 14208256 IC50 > 40000 nM T05849 CLMD93 14208257 IC50 > 40000 nM T05849 CA8ON0 14208258 IC50 = 9400 nM T05849 CXND36 14208259 IC50 = 550 nM T05849 C9YEC6 14208260 IC50 = 36000 nM T05849 CDK6O7 14208261 IC50 = 80000 nM T05849 CT14KZ 14208262 IC50 > 100000 nM T05849 C1IDH6 14208263 IC50 > 100000 nM T05849 C84QFK 14208264 IC50 = 40000 nM T05849 C1J7OL 14208265 IC50 = 180000 nM T05849 C7U4EF 14208266 IC50 = 31000 nM T05849 CC6Q1J 14208267 IC50 = 22000 nM T05849 CEK7X0 14208268 IC50 = 1900 nM T05849 C3KC0H 14208269 IC50 = 800 nM T05849 CD7M8S 14208270 IC50 = 2400 nM T05849 CU0R4P 14208271 IC50 = 1800 nM T05849 C81RHA 14208272 IC50 = 440 nM T05849 C2AC0G 14208273 IC50 = 60000 nM T05849 CU8DT5 14208274 IC50 = 6400 nM T05849 C5Q4LT 14208275 IC50 = 2400 nM T05849 CQS07B 14208280 IC50 = 73000 nM T05849 C6V0OH 14208282 IC50 = 130000 nM T05849 CP2AD3 14208283 IC50 > 100000 nM T05849 C8IAW7 14208284 IC50 = 1500 nM T05849 C4AFQ0 14208286 IC50 = 180 nM T05849 CJ63WK 14208288 IC50 = 13000 nM T05849 C3IGO6 14208293 IC50 = 750 nM T05849 CU5OL2 14208295 IC50 = 680 nM T05849 CC1NM2 14208297 IC50 = 530 nM T05849 CO4YF7 14208299 IC50 = 19000 nM T05849 CTIB05 14208300 IC50 = 5800 nM T05849 CGN9B4 14208302 IC50 = 9000 nM T05849 C7WR8Z 14208303 IC50 = 390 nM T05849 CNI38M 14208305 IC50 = 2000 nM T05849 CNV32K 14208307 IC50 = 11000 nM T05849 CWDF64 14208308 IC50 = 4400 nM T05849 C61CHZ 14208309 IC50 > 100000 nM T05849 C8MK0S 14208310 IC50 > 100000 nM T05849 C9JB4Q 14208312 IC50 = 6200 nM T05849 C2X1WI 14208313 IC50 = 3300 nM T05849 COR29A 14208315 IC50 = 38000 nM T05849 CQDF03 14208317 IC50 = 3700 nM T05849 C9WQF0 14423345 IC50 > 100000 nM T05849 CMK50F 14444002 IC50 = 5000 nM T05849 C7E6KY 14444006 IC50 = 5000 nM T05849 CYIM57 14444011 IC50 = 10000 nM T05849 CH9X8N 14444013 IC50 = 100000 nM T05849 CDG86F 14444015 IC50 = 1000 nM T05849 C1QZ0D 14444018 IC50 = 750 nM T05849 C2I3TF 14444021 IC50 = 1500 nM T05849 CZE20T 14444022 IC50 = 2000 nM T05849 CH3ER5 14444025 IC50 = 50000 nM T05849 CB64QS 14590302 IC50 > 10000 nM T05849 CQ81BH 14720386 IC50 = 7000 nM T05849 CU6KQ0 14720389 IC50 = 39000 nM T05849 CJP16B 14720390 IC50 = 17000 nM T05849 C3TJ5I 14728745 Ki = 2200 nM T05849 CI76AS 14728759 Ki = 4200 nM T05849 CRM1H2 14728761 Ki = 100000 nM T05849 CW38DZ 14728769 Ki = 580 nM T05849 C5YEL1 14728771 Ki = 1400 nM T05849 CBOQ86 14728778 Ki = 4300 nM T05849 C0B7NF 14775099 IC50 = 1400 nM T05849 C61HJW 14775102 IC50 = 1100 nM T05849 C4EVP0 14775105 IC50 = 1900 nM T05849 C3SDR6 14775108 IC50 = 1200 nM T05849 CL05HS 14775111 IC50 = 25000 nM T05849 CQTX30 14775114 IC50 = 1900 nM T05849 C65JKM 14775117 IC50 = 3400 nM T05849 CD31EJ 14776692 IC50 = 750 nM T05849 CM6E9L 14843033 IC50 = 8200 nM T05849 CL38ET 14843038 IC50 = 1300 nM T05849 C1AT3Q 14843041 IC50 = 330 nM T05849 CN0JY2 14843042 IC50 = 1600 nM T05849 CKY8S9 14991534 IC50 = 5900 nM T05849 CWSL07 14991535 IC50 = 3000 nM T05849 CNO09C 14991536 IC50 = 6100 nM T05849 CAB2I9 14991537 IC50 = 10000 nM T05849 CY0T9R 14991538 IC50 = 4800 nM T05849 C3DV5R 14991539 IC50 = 7000 nM T05849 CF7X4K 14991540 IC50 > 10000 nM T05849 CA0YW3 14991541 IC50 = 9900 nM T05849 CIS36J 14991542 IC50 = 19000 nM T05849 CO8XG9 14991543 IC50 = 10000 nM T05849 CK3I2U 14991544 IC50 = 4400 nM T05849 CASL56 14991564 IC50 = 480 nM T05849 CV3A1B 14991565 IC50 > 10000 nM T05849 CTA59E 14991566 IC50 = 10000 nM T05849 COR3I9 14991567 IC50 = 4300 nM T05849 CS87TG 14991568 IC50 = 2700 nM T05849 C51LDQ 14991569 IC50 = 1200 nM T05849 CE12JZ 14991570 IC50 = 300 nM T05849 CJFX78 14991571 IC50 = 1400 nM T05849 CCX52A 14991572 IC50 = 200 nM T05849 CDA02J 14991574 IC50 = 2100 nM T05849 C8Z0VN 14991575 IC50 = 830 nM T05849 C7LH3F 14991576 IC50 = 3000 nM T05849 CMS9P7 14991577 IC50 = 5200 nM T05849 CS9VQ1 14991578 IC50 = 87 nM T05849 CW87VU 14991579 IC50 = 4700 nM T05849 C2V7OU 14991580 IC50 = 840 nM T05849 C6L4NY 14991581 IC50 = 3600 nM T05849 CK30YF 14991582 IC50 = 3000 nM T05849 CO2MV6 14991584 IC50 = 730 nM T05849 C3VN4Q 14991585 IC50 = 570 nM T05849 CNX97Z 14991586 IC50 = 120 nM T05849 CZM0I7 15104594 IC50 = 12000 nM T05849 CH1PG7 15104595 IC50 = 7400 nM T05849 C54BNJ 15104597 IC50 > 10000 nM T05849 C9R0GF 15104598 IC50 = 27000 nM T05849 CR6C1K 15104599 IC50 > 10000 nM T05849 C3GBK1 15104600 IC50 > 10000 nM T05849 CDT0X9 15104601 IC50 = 8000 nM T05849 C0EH8B 15104602 IC50 = 3100 nM T05849 C6V5UY 15104603 IC50 > 10000 nM T05849 C58QHS 15104604 IC50 > 10000 nM T05849 CC0SN8 15104605 IC50 > 10000 nM T05849 CR6BS3 15104606 IC50 = 11000 nM T05849 CJ6N7Z 15104607 IC50 = 9700 nM T05849 C8HE4G 15104608 IC50 > 10000 nM T05849 C8MG0Q 15104609 IC50 > 10000 nM T05849 CLRX50 15104610 IC50 > 10000 nM T05849 CZR4A8 15104611 IC50 = 3300 nM T05849 CZ7TD1 15104612 IC50 > 10000 nM T05849 C6S8ZD 15104613 IC50 = 20000 nM T05849 CLJ98Q 15104615 IC50 > 10000 nM T05849 C8SRB2 15104617 IC50 > 10000 nM T05849 CO7U4V 15104618 IC50 = 5600 nM T05849 C58VEK 15104619 IC50 > 10000 nM T05849 C8TDL6 15104620 IC50 = 1900 nM T05849 CAW6C5 15104621 IC50 = 9250 nM T05849 CQ75KP 15104622 IC50 > 10000 nM T05849 CS74EB 15104623 IC50 > 10000 nM T05849 C54PSN 15104624 IC50 = 4100 nM T05849 CZ0E5N 15104625 IC50 > 10000 nM T05849 CZF98E 15104626 IC50 > 10000 nM T05849 CMD78S 15104627 IC50 = 10000 nM T05849 CBUC26 15104628 IC50 = 9200 nM T05849 C6YF2R 15104630 IC50 > 10000 nM T05849 CNT28P 15104632 IC50 > 10000 nM T05849 C4QZ6G 15167770 IC50 = 28000 nM T05849 CDGS87 15167771 IC50 > 100000 nM T05849 C7YQR1 15167772 IC50 > 100000 nM T05849 C7EN8M 15167773 IC50 > 100000 nM T05849 C62MIU 15167775 IC50 > 100000 nM T05849 CH96BN 15167776 IC50 = 5000 nM T05849 C7O4NA 15167780 IC50 > 100000 nM T05849 CH2NL5 15167783 IC50 = 24000 nM T05849 C6NBA8 15167785 IC50 > 100000 nM T05849 CG61TH 15167787 IC50 > 100000 nM T05849 C2NVC3 15167794 IC50 > 100000 nM T05849 C0KG8P 15167795 IC50 > 100000 nM T05849 CYG0O5 15167797 IC50 = 100000 nM T05849 CS1Q9A 15167799 IC50 = 74000 nM T05849 CX56VU 15167800 IC50 = 34000 nM T05849 CF7QZ6 15167802 IC50 = 13000 nM T05849 C6QMD4 15167804 IC50 = 5800 nM T05849 C6V5XT 15167808 IC50 > 10000 nM T05849 C5LJR7 15167809 IC50 > 10000 nM T05849 C5FV4M 15167811 IC50 > 100000 nM T05849 CLN01M 15167812 IC50 = 2400 nM T05849 CGQ28U 15167816 IC50 = 3200 nM T05849 C85VWQ 15167820 IC50 = 67000 nM T05849 CP8XZ1 15167824 IC50 = 21000 nM T05849 C98DJK 15200522 IC50 = 11000 nM T05849 CZJ70V 15556550 IC50 = 38000 nM T05849 CJF0P8 15614734 IC50 = 49000 nM T05849 C27OAH 15614736 IC50 > 100000 nM T05849 CEPI49 15614737 IC50 > 100000 nM T05849 CMD48W 15614739 IC50 = 14000 nM T05849 CMU7X0 15614749 IC50 = 100000 nM T05849 CI0R9Q 15614750 IC50 = 30000 nM T05849 C5JS4I 15614752 IC50 > 100000 nM T05849 CWMK79 15614762 IC50 > 100000 nM T05849 CY10TL 15614763 IC50 > 100000 nM T05849 CFS40B 15614802 IC50 > 100000 nM T05849 CR8Z9H 15614807 IC50 = 50000 nM T05849 CW5MZ1 15614818 IC50 > 100000 nM T05849 C4Z2TH 15614820 IC50 = 58000 nM T05849 CXYZ37 15614822 IC50 > 100000 nM T05849 CDH92V 15614824 IC50 = 23000 nM T05849 CM53VH 15614826 IC50 > 100000 nM T05849 C7QS6A 15614828 IC50 = 25000 nM T05849 C5OMT9 15614830 IC50 = 25000 nM T05849 CNJ8U9 15614834 IC50 > 100000 nM T05849 CZB50L 15614835 IC50 > 100000 nM T05849 CB1CY6 15614841 IC50 = 13000 nM T05849 CP6IX0 15614847 IC50 > 100000 nM T05849 C0WI1E 15614848 IC50 > 100000 nM T05849 C64JWS 15614850 IC50 > 100000 nM T05849 CY52HT 15614851 IC50 > 100000 nM T05849 CI06RY 15637150 IC50 > 100000 nM T05849 CUJ4L5 15637181 IC50 = 410 nM T05849 CD3B0H 15637183 IC50 = 300 nM T05849 C7NBP0 15637194 IC50 > 100000 nM T05849 CH6G7B 15637206 IC50 = 6.69 nM T05849 CB40AS 15666987 IC50 = 7.9 nM T05849 CS4WQ9 15666988 IC50 = 0.5 nM T05849 C5I4LT 15667001 IC50 = 140 nM T05849 CDJF92 15667003 IC50 = 0.3 nM T05849 CXH92N 15667011 IC50 = 10 nM T05849 CHK6O5 15667012 IC50 = 1.4 nM T05849 C8FOJ2 15667013 IC50 = 3.4 nM T05849 CYA7D1 15667014 IC50 = 0.59 nM T05849 CHR57O 15667015 IC50 = 24 nM T05849 CY5QE8 15667016 IC50 = 3.1 nM T05849 CD47HF 15667017 IC50 = 7.7 nM T05849 CFY0N4 15667018 IC50 = 32 nM T05849 C8P7RD 15667019 IC50 = 1.1 nM T05849 CAB7D2 15689721 IC50 = 2600 nM T05849 CVG70X 15689722 IC50 = 770 nM T05849 CS93IU 15689723 IC50 = 1600 nM T05849 CA45KS 15689724 IC50 = 3000 nM T05849 CMC0A6 15689725 IC50 = 850 nM T05849 CIX41J 15689726 IC50 = 3000 nM T05849 CD75VA 15689727 IC50 = 2600 nM T05849 C03UPY 15689728 IC50 = 7000 nM T05849 C15TYB 15689729 IC50 = 1400 nM T05849 CEC40G 15689730 IC50 = 5700 nM T05849 CRL5Z6 15689731 IC50 = 820 nM T05849 C9IF7H 15689732 IC50 = 3100 nM T05849 CFCQ31 15689733 IC50 = 1400 nM T05849 CO0FC7 15689734 IC50 = 1100 nM T05849 CSGQ09 15689735 IC50 = 2000 nM T05849 CQ08DC 15689736 IC50 = 2900 nM T05849 CQDC01 15689737 IC50 = 3700 nM T05849 C4TPD5 15689738 IC50 = 11000 nM T05849 C85PHC 15689739 IC50 = 3200 nM T05849 C5GO2B 15689740 IC50 = 2100 nM T05849 CF3R0U 15689741 IC50 = 5600 nM T05849 CRN28L 15689742 IC50 = 3300 nM T05849 CC60RH 15689743 IC50 = 1000 nM T05849 CK2EL7 15689744 IC50 = 15000 nM T05849 CTKW52 15689745 IC50 = 2000 nM T05849 C6QDI1 16090646 Ki = 501.19 nM T05849 C3UCY1 16090647 Ki < 10000 nM T05849 C3HO2S 16090649 Ki = 199.53 nM T05849 C4FKT8 16090650 Ki = 2511.89 nM T05849 CB19JY 16090651 Ki = 125.89 nM T05849 CW7KL5 16090652 Ki = 3981.07 nM T05849 C9Q5YA 16090653 Ki = 630.96 nM T05849 CA4PD3 16090658 Ki = 1584.89 nM T05849 CY9MB5 16090684 Ki = 100 nM T05849 CY91OD 16090685 Ki = 158.49 nM T05849 C4P8KS 16090686 Ki < 10000 nM T05849 C17IOA 16090687 Ki < 10000 nM T05849 C4ETX5 16090688 Ki = 316.23 nM T05849 C37DEW 16090689 Ki < 10000 nM T05849 C7Q8LP 16090690 Ki > 10000 nM T05849 COJ46W 16090691 Ki < 10000 nM T05849 CNSU17 16090692 Ki = 2511.89 nM T05849 C49PFE 16090693 Ki = 3981.07 nM T05849 CI0XC5 16090694 Ki = 31.62 nM T05849 C6QDP7 16090695 Ki = 5011.87 nM T05849 C3AVH8 16090699 Ki = 5011.87 nM T05849 C9R2PB 16090700 Ki = 1995.26 nM T05849 C9K8RC 16090701 Ki < 10000 nM T05849 CH1UB0 16090702 Ki = 1995.26 nM T05849 CD7S4Q 16090703 Ki > 10000 nM T05849 CT51EV 16090772 Ki > 10000 nM T05849 CRS7B1 16090773 Ki < 10000 nM T05849 C2KCS0 16090774 Ki < 10000 nM T05849 C8IGT2 16090780 Ki = 100 nM T05849 CM72TB 16090781 Ki = 39.81 nM T05849 C9QGU2 16090783 Ki < 10000 nM T05849 CF2IW8 16090784 Ki = 794.33 nM T05849 CKCX80 16090785 Ki > 10000 nM T05849 C3D8HU 16090786 Ki < 10000 nM T05849 C8WSC9 16090788 Ki = 158.49 nM T05849 CYQP41 16090789 Ki = 7943.28 nM T05849 C6MV4D 16090790 Ki = 15.85 nM T05849 CJ94QO 16090791 Ki = 2511.89 nM T05849 C2G8TD 16090792 Ki = 1584.89 nM T05849 CRF40D 16090793 Ki > 10000 nM T05849 CX68OS 16090794 Ki > 10000 nM T05849 C0V8WI 16090795 Ki = 1000 nM T05849 C06QBM 16090796 Ki = 1258.93 nM T05849 C5NER1 16090797 Ki = 63.1 nM T05849 C3T9MH 16100406 Ki = 1100 nM T05849 CH6F0V 16100408 Ki > 10000 nM T05849 CY5F4S 16162108 EC50 = 0.4571 nM T05849 C7YG3M 16731537 Ki = 6.026 nM T05849 C7U3FA 16731711 Ki = 23.99 nM T05849 C3G0VB 16731712 Ki = 1202.26 nM T05849 CD9KY3 16731870 Ki = 20.42 nM T05849 CMN7U9 16731871 Ki = 489.78 nM T05849 C6RS1M 16731872 Ki = 1 nM T05849 CQ45MJ 16731874 Ki = 1.862 nM T05849 C8FH9C 16732017 Ki = 1.072 nM T05849 C9I7PZ 16732018 Ki = 5.495 nM T05849 C8JR5Q 16732019 Ki = 1 nM T05849 C2OQ0S 16732020 Ki = 1.95 nM T05849 C5VUZ7 16732021 Ki = 0.7079 nM T05849 CXN1C3 16732022 Ki = 0.6607 nM T05849 C34EYO 16732162 Ki = 0.2455 nM T05849 C6CF0K 16732163 Ki = 0.2818 nM T05849 C4GZY1 16732164 Ki = 0.2951 nM T05849 C8DU5M 16732165 Ki = 0.7762 nM T05849 CB7X3W 16732442 Ki = 23.99 nM T05849 CY57CK 16732443 Ki = 4.786 nM T05849 CO95FT 16732444 Ki = 0.8318 nM T05849 CE9M8H 16732592 Ki = 9.333 nM T05849 C3J2CB 16732593 Ki = 2.754 nM T05849 CU2FT3 16732598 Ki = 331.13 nM T05849 CFT09X 16732750 Ki = 16.22 nM T05849 CM4P7G 16732753 Ki = 7.586 nM T05849 C9K4UR 16732755 Ki = 0.7943 nM T05849 CB2JR3 16732909 Ki = 2.138 nM T05849 CZ14YT 16732911 Ki = 0.6457 nM T05849 C35MZK 16732916 Ki = 5.623 nM T05849 CR0A7J 16733051 Ki = 3.89 nM T05849 C3LUI7 16733057 Ki = 4.266 nM T05849 C9FU1Q 16733182 Ki = 4.677 nM T05849 C93FYR 16733185 Ki = 1.585 nM T05849 CF3I5J 16733307 Ki = 0.3631 nM T05849 CCB36O 16733310 Ki = 0.912 nM T05849 CUF2R0 16733462 Ki = 6.166 nM T05849 C0RH7Y 16733466 Ki = 0.3388 nM T05849 C1XWA0 16733469 Ki = 0.3311 nM T05849 CK04YG 16733644 Ki = 4.074 nM T05849 C1RC2P 16733790 Ki = 16.98 nM T05849 C76HVW 16755781 IC50 > 10000 nM T05849 C5ZH6O 18656022 IC50 = 0.78 nM T05849 CX6S9T 18656023 IC50 = 0.73 nM T05849 C62KGI 18957759 IC50 = 0.59 nM T05849 CN3JW4 18957789 IC50 = 0.3 nM T05849 CMU9J5 19018661 IC50 = 4.9 nM T05849 CCNF34 19018662 IC50 = 2.7 nM T05849 CED9L0 19043358 Ki = 954.99 nM T05849 C8G1KQ 19043361 Ki = 1584.89 nM T05849 CWLN98 19043395 Ki = 954.99 nM T05849 CO64UT 19043400 Ki = 1.549 nM T05849 CCU5G4 19754254 IC50 = 72000 nM T05849 CJSH86 19754255 IC50 > 100000 nM T05849 CW3BU9 19754256 IC50 > 100000 nM T05849 C15FOQ 19754257 IC50 = 67000 nM T05849 C31FLB 19756868 IC50 = 27 nM T05849 C5WLC6 19766160 IC50 = 650 nM T05849 CNR9H0 19766161 IC50 = 17000 nM T05849 CY18ZD 19766167 IC50 = 160 nM T05849 CC0WZ1 19766168 IC50 = 2500 nM T05849 CAY89R 19766169 IC50 = 120 nM T05849 CW4Z2M 19766170 IC50 = 8600 nM T05849 C2G7OC 19766220 IC50 > 100000 nM T05849 C2ZMP1 19766221 IC50 = 38600 nM T05849 C3SL1E 19766222 IC50 > 100000 nM T05849 C6TJB9 19766227 IC50 > 100000 nM T05849 C6H9CP 19766230 IC50 > 100000 nM T05849 CNTV73 19766234 IC50 = 100000 nM T05849 CIK5L1 19910130 IC50 = 700 nM T05849 CHU7C4 20063212 IC50 = 14000 nM T05849 CF3YW5 20063240 IC50 > 100000 nM T05849 C0PGU6 20063245 IC50 = 100000 nM T05849 C5J2SZ 20063261 IC50 = 267 nM T05849 CM18EN 20190195 IC50 > 100000 nM T05849 CVF3D5 20190196 IC50 = 100000 nM T05849 C7CZ3G 20190197 IC50 = 37400 nM T05849 C8O6FN 21120982 EC50 = 13.5 nM T05849 CYG49N 21121108 IC50 = 1000 nM T05849 CK6E5Z 21246577 IC50 = 130000 nM T05849 CNH94V 21467078 IC50 = 9.8 nM T05849 CE06IA 21476261 Ki = 5.623 nM T05849 C6IE7G 21842392 IC50 = 0.1 nM T05849 CJ0YC6 23129945 IC50 = 6300 nM T05849 CDX5M1 24755148 Ki = 501.19 nM T05849 CC8IW7 24861060 IC50 > 10000 nM T05849 CZ9AS2 24861113 IC50 > 10000 nM T05849 C6TM1P 24861114 IC50 > 10000 nM T05849 CM0Q9T 24861391 IC50 > 10000 nM T05849 CA5WE4 24861392 IC50 > 10000 nM T05849 CCN34R 24861394 IC50 > 10000 nM T05849 C6YA0V 24983506 Ki = 5011.87 nM T05849 C8HMZ0 25032312 Ki < 10000 nM T05849 C3NGL2 25032468 Ki = 794.33 nM T05849 CK96SR 25033064 Ki = 1995.26 nM T05849 CM2Z9H 25033065 Ki = 5011.87 nM T05849 C1O7NJ 25033066 Ki = 1584.89 nM T05849 CITF86 25033148 Ki = 79.43 nM T05849 C67SOQ 25033149 Ki = 3162.28 nM T05849 CJ10TY 25033150 Ki = 794.33 nM T05849 C5VM9D 25033153 Ki = 1584.89 nM T05849 C5DRL8 25033224 Ki = 630.96 nM T05849 CW8C3A 25033225 Ki = 794.33 nM T05849 CVE3R2 25033226 Ki = 5011.87 nM T05849 CE6Z8Q 25033227 Ki = 1584.89 nM T05849 CR64FQ 25033229 Ki = 2511.89 nM T05849 CFBG53 25033305 Ki = 3162.28 nM T05849 CWS8F9 25033306 Ki = 3162.28 nM T05849 C6GV7F 25033307 Ki = 3981.07 nM T05849 C09CFH 25033309 Ki = 5011.87 nM T05849 C4XI0Y 25033310 Ki = 5011.87 nM T05849 CQ34SZ 25033380 Ki = 501.19 nM T05849 CN85CB 25033382 Ki = 7943.28 nM T05849 C32CSK 25033383 Ki = 7943.28 nM T05849 C43ZDF 25033384 Ki = 7943.28 nM T05849 CE1D6C 25193919 Ki = 0.021 nM T05849 C8IE3J 43811299 IC50 = 3.8 nM T05849 C2LCN6 44153340 IC50 > 100000 nM T05849 C6YES8 44209151 IC50 = 14000 nM T05849 CB6RG8 44209152 IC50 > 100000 nM T05849 CK0S6U 44209154 IC50 = 35000 nM T05849 CIZ5K3 44210424 IC50 = 18 nM T05849 CDRB36 44210425 IC50 = 270 nM T05849 CS16DE 44210426 IC50 = 5000 nM T05849 CL2P7J 44210427 IC50 = 150 nM T05849 CL7O6E 44210428 IC50 = 5400 nM T05849 CSM90K 44210535 IC50 = 1.4 nM T05849 CPH17B 44210536 IC50 = 0.36 nM T05849 C3ZK8B 44211353 IC50 = 2800 nM T05849 CZ4YJ5 44211354 IC50 = 600 nM T05849 C0K6XC 44212230 Ki = 7.586 nM T05849 CAO2M3 44212546 IC50 = 12 nM T05849 C19WBD 44215880 Ki = 15300 nM T05849 C4M2QS 44271859 Ki = 301 nM T05849 C2UFZ4 44271963 Ki = 0.56 nM T05849 C8K4UV 44272041 Ki = 9.11 nM T05849 C31VQG 44272042 Ki = 29.2 nM T05849 C23PKL 44272076 Ki = 4.7 nM T05849 CH1KX2 44272156 Ki = 27.5 nM T05849 C2KM5N 44279808 IC50 = 370 nM T05849 CDUE85 44279809 IC50 = 110 nM T05849 C5J9IA 44279810 IC50 = 115 nM T05849 C5JGZ1 44279811 IC50 = 136 nM T05849 C8J6ZD 44279852 IC50 = 206 nM T05849 CJKP43 44279853 IC50 = 142 nM T05849 CORN87 44279861 IC50 = 80 nM T05849 CA21WF 44279862 IC50 = 570 nM T05849 C1IKY0 44279937 IC50 = 37 nM T05849 C14KNC 44279938 IC50 = 24 nM T05849 CDQ3P2 44279939 IC50 = 9 nM T05849 CFR9C4 44279957 IC50 = 51 nM T05849 C2XHW4 44279985 IC50 = 1252 nM T05849 CPNG71 44280000 IC50 = 600 nM T05849 C5N1VJ 44280028 IC50 = 45 nM T05849 C0CSF5 44280029 IC50 = 240 nM T05849 CT6ZV8 44280090 IC50 = 13 nM T05849 CXE4S2 44280091 IC50 = 51 nM T05849 CO9VU0 44280101 IC50 = 97 nM T05849 C1B9HX 44280102 IC50 = 55 nM T05849 CNE5U3 44280103 IC50 = 54 nM T05849 C79ZUL 44280110 IC50 = 241 nM T05849 CF68MD 44280111 IC50 = 49 nM T05849 C0N3WK 44280112 IC50 = 25 nM T05849 CXM89F 44280113 IC50 = 118 nM T05849 C8SFO2 44280114 IC50 = 3400 nM T05849 CEWR83 44280115 IC50 = 550 nM T05849 C92DXF 44280116 IC50 = 230 nM T05849 C12TGJ 44280117 IC50 = 155 nM T05849 C3LS7R 44280122 IC50 = 57 nM T05849 CPC5D3 44280123 IC50 = 216 nM T05849 CBYO06 44280130 IC50 = 26 nM T05849 C26NSK 44280131 IC50 = 19 nM T05849 CQ2DB5 44280163 IC50 = 27 nM T05849 CTF0M6 44280176 IC50 = 86 nM T05849 CJ0C2S 44280177 IC50 = 343 nM T05849 CMVA74 44280178 IC50 = 31 nM T05849 C3S2ZJ 44280179 IC50 = 126 nM T05849 CL3F8R 44280180 IC50 = 168 nM T05849 CM4OD6 44280193 IC50 = 101 nM T05849 CMZH06 44280200 IC50 = 16 nM T05849 CUEZ53 44280205 IC50 = 76 nM T05849 CU3V7K 44280213 IC50 = 135 nM T05849 C6XP3Y 44280214 IC50 = 14 nM T05849 C47YAI 44280215 IC50 = 25 nM T05849 CS71DY 44280224 IC50 = 210 nM T05849 CD6CA5 44280225 IC50 = 185 nM T05849 C6MJ3B 44280233 IC50 = 37 nM T05849 CJ87NF 44280234 IC50 = 38 nM T05849 CAOP30 44280244 IC50 = 54 nM T05849 C81HWG 44280245 IC50 = 13 nM T05849 CWAS89 44280246 IC50 = 32 nM T05849 CH71DF 44280252 IC50 = 3 nM T05849 C7MY4S 44280266 IC50 = 790 nM T05849 CTI89O 44280269 IC50 = 9 nM T05849 C6WQL5 44280270 IC50 = 82 nM T05849 CB2TG3 44280314 IC50 = 12 nM T05849 C1SXP7 44280315 IC50 = 55 nM T05849 CV2C8I 44280316 IC50 = 23 nM T05849 C3NV9D 44280350 IC50 = 44 nM T05849 C41WEC 44280363 IC50 = 2810 nM T05849 C4M5YT 44280368 IC50 = 1083 nM T05849 CEN48R 44280371 IC50 = 32 nM T05849 CB08JV 44280372 IC50 = 60 nM T05849 C3EUS8 44280373 IC50 = 200 nM T05849 CE3NV9 44280374 IC50 = 161 nM T05849 C7DR5X 44280375 IC50 = 568 nM T05849 CPS32U 44280380 IC50 = 95 nM T05849 CS2ET3 44280381 IC50 = 488 nM T05849 C8IH4X 44280387 IC50 = 443 nM T05849 CZ76BA 44280388 IC50 = 63 nM T05849 C9YQ4P 44280397 IC50 = 36 nM T05849 CU3W4Q 44280398 IC50 = 71 nM T05849 C6T0HX 44280399 IC50 = 173 nM T05849 CLQ6R7 44280406 IC50 = 166 nM T05849 C0KBA8 44280407 IC50 = 9 nM T05849 C4H2UP 44280414 IC50 = 63 nM T05849 CUE5P2 44280495 IC50 = 380 nM T05849 C9L7UJ 44280501 IC50 = 9 nM T05849 CO13XU 44280502 IC50 = 398 nM T05849 C2U1BA 44280507 IC50 = 80 nM T05849 CZ6M2H 44280508 IC50 = 75 nM T05849 CV85OR 44280509 IC50 = 155 nM T05849 C2DCL5 44280510 IC50 = 162 nM T05849 CF0W6B 44280598 IC50 = 17 nM T05849 CL1CG4 44280599 IC50 = 7 nM T05849 C3P2UJ 44280620 IC50 = 117 nM T05849 CG3M0X 44280621 IC50 = 57 nM T05849 CE8QZ1 44280622 IC50 = 16 nM T05849 CAI7D3 44280694 IC50 = 316 nM T05849 CA3C2F 44280713 IC50 = 190 nM T05849 CMYG13 44280714 IC50 = 75 nM T05849 CH94XP 44280729 IC50 = 76 nM T05849 CWU8C9 44280740 IC50 = 23 nM T05849 CQ05TE 44280741 IC50 = 36 nM T05849 C15PNE 44280893 IC50 = 233 nM T05849 CNZS40 44280894 IC50 = 48 nM T05849 CP6K3O 44280895 IC50 = 119 nM T05849 C2XUO4 44280915 IC50 = 1351 nM T05849 CE5Z1T 44280973 IC50 = 89 nM T05849 CZ5MW8 44280974 IC50 = 185 nM T05849 CPZ8U2 44280992 IC50 = 114 nM T05849 C72TIJ 44280993 IC50 = 691 nM T05849 CR8LE1 44280996 IC50 = 11 nM T05849 CLB35W 44281004 IC50 = 220 nM T05849 CXQ4J5 44281005 IC50 = 135 nM T05849 CP3K5O 44281020 IC50 = 26 nM T05849 CL70PJ 44281078 IC50 = 27 nM T05849 CMWH08 44281084 IC50 = 1017 nM T05849 C5RUZ7 44281204 IC50 = 9 nM T05849 CGEB47 44281205 IC50 = 7 nM T05849 CG67IC 44281292 IC50 = 19 nM T05849 CC9W7Y 44283580 IC50 > 10000 nM T05849 CSOQ87 44283602 IC50 = 4000 nM T05849 C13DXZ 44283660 IC50 = 7000 nM T05849 CGHY18 44283873 IC50 > 10000 nM T05849 CH6IU4 44286379 IC50 = 22700 nM T05849 C5GF2B 44293810 IC50 = 0.47 nM T05849 CT9NI7 44293811 IC50 = 2 nM T05849 CL85QH 44293812 IC50 = 1.8 nM T05849 C5OAG3 44293892 IC50 = 0.37 nM T05849 CY40KR 44293971 IC50 = 0.96 nM T05849 CEH10G 44293998 IC50 = 0.84 nM T05849 CV13IT 44293999 IC50 = 1 nM T05849 C7DUC8 44300550 IC50 = 29.9 nM T05849 C5DA9R 44300551 IC50 = 16 nM T05849 C3O6HU 44300743 IC50 = 0.22 nM T05849 CT5RZ1 44300744 IC50 = 2.7 nM T05849 C8EK9U 44300745 IC50 = 0.6 nM T05849 CY1FN6 44300852 IC50 = 0.81 nM T05849 CPHZ41 44300862 IC50 = 4.2 nM T05849 CFW7D1 44300863 IC50 = 0.88 nM T05849 CG5LP1 44300864 IC50 = 4.8 nM T05849 CQ74BL 44300888 IC50 = 9 nM T05849 C8KOW2 44300889 IC50 = 0.98 nM T05849 C0Y2QV 44300890 IC50 = 1.7 nM T05849 CGEA85 44300891 IC50 = 0.88 nM T05849 CP3OK7 44300989 IC50 = 0.26 nM T05849 C7GY2R 44301015 IC50 = 0.7 nM T05849 CF0R7T 44301016 IC50 = 5.1 nM T05849 CGMT91 44301034 IC50 = 1.4 nM T05849 CZB0W1 44301036 IC50 = 7.9 nM T05849 CBMY25 44301037 IC50 = 1 nM T05849 CO59MI 44303224 IC50 = 1000 nM T05849 C6J7EK 44303510 IC50 = 4528 nM T05849 CWKM16 44303511 IC50 = 1881 nM T05849 CY5Q8R 44303654 IC50 = 169 nM T05849 CNH0W1 44303663 IC50 > 10000 nM T05849 CD80VI 44303664 IC50 = 1.9 nM T05849 C0L8GD 44303722 IC50 = 4251 nM T05849 C1VM8Q 44306360 IC50 = 100000 nM T05849 C3ZDK0 44306744 IC50 = 5011.87 nM T05849 CB5Q6O 44306823 IC50 = 1000 nM T05849 CG9HF2 44306868 IC50 = 63095.73 nM T05849 CP92WE 44306887 IC50 = 50118.72 nM T05849 CN0SR5 44306888 IC50 = 10000 nM T05849 C81TNA 44309988 IC50 > 100000 nM T05849 CGE4Q1 44311593 IC50 > 10000 nM T05849 C05ZPL 44311626 IC50 > 100000 nM T05849 C5N7QT 44311642 IC50 > 10000 nM T05849 CBFJ81 44311923 IC50 = 7000 nM T05849 CCE47R 44311939 IC50 = 1200 nM T05849 C2K5WT 44311988 IC50 = 55000 nM T05849 CHP0A5 44312020 IC50 > 100000 nM T05849 CW5JD6 44312041 IC50 > 100000 nM T05849 CER8O2 44313549 IC50 = 0.24 nM T05849 CE2K0Q 44318205 IC50 = 2.4 nM T05849 COS38V 44318234 IC50 = 18 nM T05849 C4RBF2 44318341 Ki = 0.4 nM T05849 COAF14 44327225 EC50 = 6 nM T05849 CPAX62 44327502 EC50 = 12 nM T05849 CXB5P4 44327506 EC50 = 19 nM T05849 C92SBQ 44327526 EC50 = 265 nM T05849 CZS19I 44327580 EC50 = 9 nM T05849 CYXH20 44327581 EC50 = 140 nM T05849 C3MR8J 44328894 Ki = 0.3981 nM T05849 C10ORA 44328951 Ki = 12.59 nM T05849 CY68ZI 44329055 IC50 = 25 nM T05849 CP3I1N 44329150 IC50 = 134 nM T05849 CZFL34 44329156 Ki = 1.585 nM T05849 C5H7YJ 44329286 IC50 = 66 nM T05849 C6R7XF 44329287 IC50 = 65 nM T05849 C7HBW4 44329304 IC50 = 80 nM T05849 CJ91PD 44329305 IC50 = 453 nM T05849 C4GRP3 44329306 IC50 = 38 nM T05849 CYB43Q 44329323 IC50 = 71 nM T05849 C7UCB1 44329324 IC50 = 278 nM T05849 CHC5O3 44329325 IC50 = 79 nM T05849 CQFK89 44329330 IC50 = 141 nM T05849 C8EZS5 44329331 IC50 = 190 nM T05849 C6TE7J 44329342 IC50 = 10 nM T05849 CYL34Q 44329343 IC50 = 87 nM T05849 C05TEI 44329352 IC50 = 36 nM T05849 CRFX63 44329363 IC50 = 28 nM T05849 C2Q5IU 44329383 IC50 = 450 nM T05849 CMVE80 44329384 IC50 = 28 nM T05849 C1FU0W 44329398 Ki = 224 nM T05849 CF5E7K 44329442 IC50 = 560 nM T05849 CHA59U 44329456 IC50 = 16 nM T05849 CX30GP 44329486 IC50 = 203 nM T05849 C65UFJ 44329487 IC50 = 31 nM T05849 C17ETM 44329518 IC50 = 117 nM T05849 CVO8J6 44329519 IC50 = 28 nM T05849 C43HSM 44329520 IC50 = 40 nM T05849 CZH8V1 44329798 Ki = 12.3 nM T05849 CORU67 44330731 IC50 = 15 nM T05849 CT7I5W 44330874 IC50 = 8.7 nM T05849 C5PV3J 44331065 IC50 = 16 nM T05849 C3MQS5 44331343 Ki = 34.67 nM T05849 C6SE3Q 44331431 IC50 = 1900 nM T05849 CN43PT 44331467 Ki = 33.88 nM T05849 C4F7CG 44331468 Ki = 3.89 nM T05849 CH2W6E 44331479 Ki = 28.84 nM T05849 CBA7U5 44331483 Ki = 42.66 nM T05849 CU5MC4 44331489 Ki = 2.57 nM T05849 C4KNX0 44331505 Ki = 2.399 nM T05849 C3OL4H 44331506 Ki = 10.72 nM T05849 CEI8L2 44331524 Ki = 16.98 nM T05849 CJ6DO2 44332766 Ki = 223.87 nM T05849 C4ES6H 44333048 IC50 = 13 nM T05849 CG9SW2 44333049 IC50 = 2 nM T05849 CDU94X 44333078 IC50 = 7 nM T05849 C5EZD1 44333219 IC50 > 3000 nM T05849 C8CQZ6 44333278 IC50 = 31 nM T05849 C1IY3U 44333305 IC50 = 11.8 nM T05849 C2ZLD0 44333311 IC50 = 18.3 nM T05849 CT5B6W 44333312 IC50 = 880 nM T05849 CT9B6O 44333341 IC50 = 270 nM T05849 C5YAJ0 44333624 IC50 = 4.9 nM T05849 CD2C1U 44333997 IC50 = 912 nM T05849 CS2BA0 44334033 IC50 > 10000 nM T05849 CX73QJ 44334172 IC50 = 2000 nM T05849 C2L7QP 44334176 IC50 = 410 nM T05849 CF3J5W 44334177 IC50 > 6000 nM T05849 C1F6CN 44334224 IC50 = 1500 nM T05849 C9VJE6 44334225 IC50 = 180 nM T05849 C4HB5R 44334237 IC50 > 10000 nM T05849 C4ODL2 44334248 IC50 = 120 nM T05849 C0JZ5A 44334250 IC50 > 10000 nM T05849 CADP45 44334258 IC50 = 2000 nM T05849 CCW7M2 44334259 IC50 = 4800 nM T05849 CF8P4L 44334270 IC50 > 6900 nM T05849 CRUK97 44334278 IC50 = 390 nM T05849 CX42MS 44334305 IC50 = 160 nM T05849 C1J3GT 44334320 IC50 = 170 nM T05849 CX8O1B 44334325 IC50 > 5900 nM T05849 CDN23P 44334330 IC50 > 10000 nM T05849 CPD10L 44334331 IC50 > 10000 nM T05849 C69VYO 44334332 IC50 > 10000 nM T05849 C2R0EQ 44334337 IC50 = 900 nM T05849 CU53LB 44334338 IC50 = 810 nM T05849 CRI9C6 44334345 IC50 = 53 nM T05849 C3CI0L 44334354 IC50 = 230 nM T05849 C0NI9K 44334379 IC50 = 5700 nM T05849 CTK69B 44334434 IC50 = 3900 nM T05849 CF32EL 44334438 IC50 = 440 nM T05849 C45YUA 44334452 IC50 = 1100 nM T05849 CK29CZ 44334704 IC50 = 300 nM T05849 C4G1WN 44336539 IC50 = 48.6 nM T05849 C4EP8X 44341327 IC50 = 10000 nM T05849 CZ7G1F 44341426 IC50 < 10000 nM T05849 CM7NI2 44341429 IC50 = 100000 nM T05849 CCZ54K 44341613 IC50 = 7600 nM T05849 C16CFB 44345946 Ki = 3.802 nM T05849 C93LEP 44345980 Ki = 0.2884 nM T05849 CH58ZU 44346047 Ki = 0.2239 nM T05849 C64KRV 44346097 Ki = 5.248 nM T05849 C0I8TH 44346126 Ki = 1.738 nM T05849 CY8X4R 44346176 Ki = 3.548 nM T05849 C0GF4Z 44346225 Ki = 0.1778 nM T05849 CX4G1M 44346255 Ki = 1.514 nM T05849 C7G5EM 44346296 Ki = 0.955 nM T05849 C0S2CQ 44346321 Ki = 1460 nM T05849 C18CLD 44346326 Ki = 2.089 nM T05849 CR56CO 44346345 Ki = 1.023 nM T05849 C15WNJ 44346355 Ki = 6.4 nM T05849 CE42SR 44346508 Ki > 3000 nM T05849 C9F0GT 44346587 Ki = 11.9 nM T05849 CMB2N8 44346623 Ki = 4.8 nM T05849 CMVS97 44346651 Ki = 0.15 nM T05849 C5DU4C 44348808 IC50 = 23000 nM T05849 CD63MX 44349069 IC50 = 200 nM T05849 CC83MK 44349070 IC50 = 800 nM T05849 CA14VC 44349082 IC50 = 8300 nM T05849 C5T8SC 44349314 IC50 = 2000 nM T05849 CK83MG 44349383 IC50 = 8100 nM T05849 C7K0EY 44349572 IC50 = 2.2 nM T05849 CBU69Q 44351413 Ki = 775 nM T05849 CT2V3U 44351414 Ki = 122 nM T05849 C3LM0J 44351415 Ki = 56 nM T05849 CG7YT6 44351444 Ki = 6.8 nM T05849 C50XEB 44351445 Ki = 1.9 nM T05849 C5KAV7 44351446 Ki = 0.5 nM T05849 CMG73P 44351454 Ki = 44.8 nM T05849 CKP1Q5 44351455 Ki = 26.2 nM T05849 C3UTY1 44351469 Ki = 6.1 nM T05849 C6N9XA 44351477 Ki = 14 nM T05849 CI0UW3 44351491 Ki = 20 nM T05849 CWI6B0 44351492 Ki = 24 nM T05849 CE50BX 44351519 Ki = 24 nM T05849 C57NMK 44351524 Ki = 32 nM T05849 C4HYP6 44355590 Ki = 2.1 nM T05849 CVO2G3 44355745 Ki = 1.6 nM T05849 CMS4H1 44355747 Ki = 0.6 nM T05849 C8VW0Y 44355787 Ki = 2.1 nM T05849 C61FUJ 44356619 IC50 = 460 nM T05849 C60UCN 44356620 IC50 = 500 nM T05849 CJ7I2B 44356645 IC50 = 46 nM T05849 CX5L4J 44356697 IC50 = 32.6 nM T05849 CMJ78F 44356710 IC50 = 4.8 nM T05849 CFA0U2 44356717 IC50 = 170 nM T05849 C35PBX 44356726 IC50 = 26 nM T05849 C4B2DC 44356788 IC50 = 6 nM T05849 CLR4M9 44356799 IC50 = 5.7 nM T05849 CZDM24 44356801 IC50 = 22 nM T05849 C6KNQ0 44356868 IC50 = 22 nM T05849 CVA89M 44356972 IC50 = 130 nM T05849 CY3FE7 44357031 IC50 = 9.7 nM T05849 CGD1A9 44357068 IC50 = 5.9 nM T05849 C3P4EN 44357198 IC50 = 104 nM T05849 COXI10 44359484 Ki = 0.15 nM T05849 C5K6BZ 44359840 IC50 = 100000 nM T05849 C0DB9O 44359841 IC50 > 100000 nM T05849 C2M3SG 44359865 IC50 > 100000 nM T05849 C8JQD5 44359866 IC50 > 100000 nM T05849 CQC78O 44359879 IC50 > 100000 nM T05849 C3TX5W 44359880 IC50 = 100000 nM T05849 CZC76O 44359881 IC50 = 55000 nM T05849 C1U0RS 44360121 IC50 > 100000 nM T05849 CN9LB0 44360216 IC50 > 100000 nM T05849 C9X8SL 44360340 IC50 = 23000 nM T05849 CHAZ51 44365304 IC50 = 1584.89 nM T05849 CMV8Q7 44365359 IC50 = 31622.78 nM T05849 C1RNC2 44365788 IC50 = 199.53 nM T05849 C58SDA 44365965 IC50 = 2000 nM T05849 C12RAO 44365966 IC50 > 10000 nM T05849 C7P8LD 44365993 IC50 = 20000 nM T05849 CZO85D 44366097 IC50 = 30000 nM T05849 C1CQI7 44366107 IC50 = 25000 nM T05849 C2XMY6 44366108 IC50 = 15000 nM T05849 CH4Z8J 44366188 IC50 = 50000 nM T05849 C9ZY7M 44366341 IC50 = 10000 nM T05849 C2CAI4 44368454 IC50 > 100000 nM T05849 CU63DH 44370393 IC50 = 430 nM T05849 CFH0W4 44370406 IC50 = 44000 nM T05849 C1R4AQ 44370446 IC50 = 4500 nM T05849 C5GFJ8 44370451 IC50 = 310 nM T05849 CI42BZ 44370461 IC50 = 860 nM T05849 C4YTD1 44370473 IC50 = 13000 nM T05849 CO3AW8 44370497 IC50 = 4100 nM T05849 CIV24D 44370505 IC50 = 100000 nM T05849 CKXE79 44370694 IC50 = 190 nM T05849 C8RXJ1 44372047 IC50 > 10000 nM T05849 CVR3W2 44372063 IC50 = 775 nM T05849 CD0N1Y 44372201 IC50 = 3720 nM T05849 CL1B5X 44372320 IC50 > 10000 nM T05849 CUC38J 44372327 IC50 = 69200 nM T05849 CVDF90 44376112 IC50 = 1.02 nM T05849 CKL8F9 44376113 IC50 = 0.142 nM T05849 C87VGD 44376130 IC50 = 8.5 nM T05849 C1BUI3 44376132 IC50 = 23.8 nM T05849 CC71KL 44376191 IC50 = 250 nM T05849 CKLZ40 44377486 IC50 = 90 nM T05849 C3K1QN 44377487 IC50 = 81000 nM T05849 CQ4AI8 44377488 IC50 = 75000 nM T05849 C4RGT7 44377587 IC50 = 110000 nM T05849 CC91FE 44377588 IC50 = 15000 nM T05849 C6QLO5 44377589 IC50 = 6000 nM T05849 CTK59G 44377790 IC50 = 1200 nM T05849 C7WJS8 44377852 IC50 = 78000 nM T05849 CB86IA 44379188 Ki = 1.7 nM T05849 C6H0NB 44381138 Ki = 0.46 nM T05849 CBS7G0 44381201 IC50 = 1800 nM T05849 CR8IJ7 44381202 IC50 = 700 nM T05849 CJMB63 44381358 Ki = 0.06 nM T05849 CNRM40 44381463 IC50 = 53 nM T05849 CW4N8P 44381479 IC50 = 730 nM T05849 CU64YH 44381480 IC50 = 4500 nM T05849 C6QP7N 44381481 IC50 > 10000 nM T05849 C49RXM 44381482 IC50 > 10000 nM T05849 CU1IX9 44381489 IC50 = 600 nM T05849 CP0ZY4 44381513 IC50 = 72 nM T05849 COES56 44381550 IC50 = 2400 nM T05849 CGO7M8 44381562 IC50 = 2500 nM T05849 CQ9R3A 44381577 IC50 = 7000 nM T05849 C0M9AG 44381578 IC50 = 3800 nM T05849 CZT9Y8 44381593 IC50 = 5000 nM T05849 C9TP6E 44381695 IC50 = 1400 nM T05849 C17PCH 44381719 IC50 = 42200 nM T05849 CG6D5A 44381730 IC50 = 103800 nM T05849 CG13QU 44381749 IC50 = 50000 nM T05849 CU0C8S 44381758 IC50 = 3300 nM T05849 C4IKD6 44381815 IC50 = 710 nM T05849 CZH29J 44381829 IC50 = 3600 nM T05849 CTU58L 44381892 IC50 = 12500 nM T05849 C3LER5 44381914 IC50 = 16000 nM T05849 C7YA0B 44381925 IC50 = 2600 nM T05849 CAP12B 44381949 IC50 = 270 nM T05849 CR9GY4 44381960 IC50 = 5900 nM T05849 CR3U2T 44382008 IC50 = 11000 nM T05849 CS7T6K 44382038 IC50 = 109 nM T05849 C2W0DJ 44382057 IC50 = 878 nM T05849 CT1YO0 44382327 IC50 = 1190 nM T05849 C2Y7GM 44382371 IC50 = 103 nM T05849 CEP95N 44387568 Ki = 15 nM T05849 CQ1L2U 44396655 EC50 = 98 nM T05849 CLO4M3 44396745 EC50 = 517 nM T05849 C3WS6P 44396746 IC50 = 1610 nM T05849 C9TZV6 44398261 IC50 > 10000 nM T05849 CNI58U 44403829 IC50 = 136 nM T05849 CD69PS 44408411 Ki = 1700 nM T05849 C7QV6M 44408483 Ki = 930 nM T05849 C96ELC 44408632 Ki = 560 nM T05849 CI26KP 44417427 Ki = 63.1 nM T05849 C0CV9L 44417429 Ki = 100 nM T05849 CNZ3I4 44417439 Ki = 1258.93 nM T05849 C5OI3W 44418923 IC50 = 15.85 nM T05849 C4UPR1 44418924 IC50 = 4.571 nM T05849 CWT4D8 44425005 Ki = 89.13 nM T05849 C2PEJ5 44425006 Ki = 1.202 nM T05849 CKTE61 44445282 Ki = 1995.26 nM T05849 C1NPO4 44445283 Ki = 6309.57 nM T05849 CL94GA 44451519 Ki = 7.586 nM T05849 CXJ5N0 44451522 Ki = 23.44 nM T05849 CN8B5I 44451523 Ki = 380.19 nM T05849 CMF6V5 44451547 Ki = 4.266 nM T05849 C2MP5A 44451581 Ki = 0.8913 nM T05849 C9SC7M 44451622 Ki = 6.31 nM T05849 CH1K6S 44451830 Ki = 501.19 nM T05849 CWEV38 44451843 Ki = 3.162 nM T05849 CIS9D2 44451877 Ki = 9.55 nM T05849 CVN2E4 44451920 Ki = 9.55 nM T05849 CBPT84 44458049 IC50 = 4800 nM T05849 CNH24L 44458050 IC50 >> 10000 nM T05849 C5I3KT 44458068 IC50 > 10000 nM T05849 C9S5UT 44458096 IC50 = 7350 nM T05849 CF2RM4 44458101 IC50 > 10000 nM T05849 CPVM59 44458102 IC50 >> 10000 nM T05849 CV2K8W 44458112 IC50 > 10000 nM T05849 CYS0T8 44458113 IC50 > 10000 nM T05849 CIW1N6 44458114 IC50 > 10000 nM T05849 C7ONM9 44458120 IC50 = 2000 nM T05849 C94RSO 44578686 IC50 > 10000 nM T05849 CLW1R5 44578727 IC50 > 10000 nM T05849 CDIW83 44578728 IC50 > 10000 nM T05849 CCP04Y 44578729 IC50 > 10000 nM T05849 CJE1O8 44578764 IC50 > 10000 nM T05849 C2A4JT 44578767 IC50 > 10000 nM T05849 C76AQL 44580898 Ki = 3.9 nM T05849 C3S2XF 44580899 Ki = 7.3 nM T05849 C6Q3NU 44580900 Ki = 16.3 nM T05849 CSH7E8 44580901 Ki = 14.2 nM T05849 C6XOD8 44580932 Ki = 0.0407 nM T05849 C6FE1M 45102806 Ki = 10 nM T05849 CM6BH7 45255234 Ki = 15.85 nM T05849 CR3ZF1 45262813 IC50 = 1.35 nM T05849 CYTL70 45486933 Ki = 398.11 nM T05849 CQH80S 45486935 Ki = 10 nM T05849 C7YUL8 45486936 Ki = 6.31 nM T05849 C1KLB2 45486940 Ki = 63.1 nM T05849 COT6U7 45486941 Ki = 630.96 nM T05849 CAQ7Z9 45486947 Ki = 251.19 nM T05849 C6FGL0 45486949 Ki = 79.43 nM T05849 CSR39Z 45486955 Ki = 39.81 nM T05849 CDZ82O 45486958 Ki = 158.49 nM T05849 CMI20Q 45486964 Ki = 10 nM T05849 CD02XL 45486967 Ki = 6309.57 nM T05849 C1X3BW 45486968 Ki = 630.96 nM T05849 CC8W1B 45486969 Ki = 1584.89 nM T05849 CV17ZB 45486970 Ki = 1000 nM T05849 CZ04GO 45486971 Ki = 1258.93 nM T05849 C2WJI9 45486974 Ki = 1258.93 nM T05849 C5HP4B 45486976 Ki = 6.31 nM T05849 CXR7T6 45486985 Ki = 5.012 nM T05849 CIX0G1 45486994 Ki > 10000 nM T05849 C1PZ8J 45486995 Ki = 1000 nM T05849 C06PMK 45486997 Ki = 316.23 nM T05849 CQ31XM 45487002 Ki = 12.59 nM T05849 C3YB8W 45487003 Ki = 7943.28 nM T05849 C6SQZ7 45487006 Ki = 10 nM T05849 CD0WG8 46235271 Ki = 69.18 nM T05849 C94EJG 46869398 IC50 > 10000 nM T05849 C8Y2QS 49798104 IC50 = 125.89 nM T05849 C6LEM8 49798106 Ki = 930 nM T05849 C8EG6Y 49798111 Ki = 18 nM T05849 C24DUW 49798112 Ki = 120 nM T05849 CAM0I2 49798148 Ki = 61 nM T05849 CP0NO1 52950956 IC50 = 0.6 nM T05849 C7PC2V 52950958 IC50 = 0.8 nM T05849 CMYU60 52951093 IC50 = 3.6 nM T05849 C8ZL7M 52951227 IC50 = 1.6 nM T05849 C2VK4G 52951333 IC50 = 2.4 nM T05849 CG80QW 52951789 IC50 = 2.4 nM T05849 CXZL73 52952034 IC50 = 0.9 nM T05849 C6UQ3N 53233689 IC50 > 10000 nM T05849 C2DIE0 53465843 Ki = 1000 nM T05849 CB90RU 53465844 Ki = 1000 nM T05849 C4HMO9 56663037 IC50 = 4.8 nM T05849 CZL6U4 56663263 IC50 = 2.5 nM T05849 CRL92U 56666696 IC50 = 3.4 nM T05849 CV38BZ 56683899 IC50 = 0.7 nM T05849 CLS4N8 57390472 IC50 = 450 nM T05849 CD4B1K 57392083 Ki = 3100 nM T05849 CQ92LO 57393204 IC50 = 420 nM T05849 CM4SX5 57394919 IC50 > 100000 nM T05849 C4UPK7 57395574 Ki = 18000 nM T05849 CUIC13 70684970 IC50 = 140000 nM T05849 CYD85N 70687140 IC50 > 100000 nM T05849 C0L3SF 70689205 IC50 > 100000 nM T05849 C89CIK 70697518 IC50 = 100000 nM T05849 CFKB17 70697534 IC50 = 18000 nM T05849 CRI31Z 71449099 IC50 = 19 nM T05849 C1HA5U 71452639 IC50 > 10000 nM T05849 C2EDN7 71580808 IC50 = 16 nM T05849 C43WGZ 71717880 IC50 = 0.9 nM T05849 C3XJ9W 73345199 IC50 = 1400 nM T05849 C5G9XQ 73345482 Ki = 120 nM T05849 C62DYB 73345878 IC50 = 4600000 nM T05849 CCUJ79 73346731 IC50 = 32 nM T05849 CM76NZ 73346732 IC50 = 1200 nM T05849 C5KT3R 73346888 IC50 = 3981.07 nM T05849 C3A4YR 73347063 Ki = 15 nM T05849 C2HY0X 73347220 Ki = 1 nM T05849 C8P9WM 73347384 IC50 = 6 nM T05849 C0DT6B 73348733 Ki = 0.13 nM T05849 CQ1ME6 73349806 IC50 = 57 nM T05849 CBC73K 73349808 IC50 = 1800 nM T05849 C7VX8Q 73350067 EC50 = 54 nM T05849 CE9L2I 73350093 Ki = 6.43 nM T05849 C3IN9K 73350475 IC50 = 8.5 nM T05849 C3QUR8 73351326 IC50 = 190 nM T05849 CFG96R 73351327 IC50 = 200 nM T05849 CRO1M7 73351812 Ki = 0.8 nM T05849 C8PL7I 73351992 IC50 = 5.2 nM T05849 COE81N 73353042 Ki = 290 nM T05849 C6XW5D 73353455 IC50 = 12 nM T05849 CU0ZM1 73354298 IC50 = 1150 nM T05849 CM93DB 73354642 Ki = 62 nM T05849 CA8MQ1 73354785 IC50 = 199.53 nM T05849 CMQW89 90663193 IC50 = 25 nM T05849 CNF64R 90663239 EC50 = 80 nM T05849 C05KGQ 90663271 IC50 = 1.9 nM T05849 C8KP9Y 90663974 IC50 = 730 nM T05849 CK8U0X 90663975 IC50 = 970 nM T05849 C0U7FK 90663976 IC50 = 210 nM T05849 CU5D2N 90663977 IC50 = 1800 nM T05849 C21HNI 90663978 IC50 = 3000 nM T05849 CZ26FG 90663979 IC50 = 4000 nM T05849 CR7S3I 90663980 IC50 = 5000 nM T05849 C96MAN 90663981 IC50 = 5000 nM T05849 C8H9MP 90663982 IC50 = 750 nM T05849 COAU27 90663983 IC50 = 5300 nM T05849 C3ZJ5B 90663984 IC50 = 1700 nM T05849 C3SWD6 90663985 IC50 = 1700 nM T05849 C1BS3K 90663986 IC50 = 2900 nM T05849 CE0KD8 90663991 IC50 = 4400 nM T05849 CMP96Z 90663992 IC50 = 2100 nM T05849 C2I8VH 90663993 IC50 = 5100 nM T05849 C1VBU5 90663994 IC50 = 1500 nM T05849 CW6PS8 90663995 IC50 = 470 nM T05849 C08XBU 90663996 IC50 = 238 nM T05849 C45ZPT 101918113 IC50 = 70 nM T05849 C6SL9D 118718805 IC50 > 100000 nM T05849 CT2U5K 118718843 Ki = 3.2 nM T05849 CGZ8P7 118719062 Ki = 93 nM T05849 C63VPI 118719097 Ki = 54 nM T05849 CI7ZL6 118719276 Ki = 590 nM T05849 CEZ7C1 118719277 Ki = 3000 nM T05849 C4XI9Q 118719278 Ki = 71 nM T05849 C4A3NV 118719279 Ki = 68 nM T05849 C3X7BR 118719280 Ki = 140 nM T05849 CC8UQ7 118719281 Ki = 2.8 nM T05849 CW7BG8 118719282 Ki = 5.1 nM T05849 CPKM62 118719283 Ki = 14 nM T05849 C10SUD 118719284 Ki = 74 nM T05849 CAB7P9 118719285 Ki = 39 nM T05849 C4DB3S 118719286 Ki = 17 nM T05849 CMN98J 118719287 Ki = 81 nM T05849 CL6AC9 118719288 Ki = 170 nM T05849 CV8KN7 118719289 Ki = 770 nM T05849 C9FM5Q 118719290 Ki = 36 nM T05849 CA7HE8 118727696 Ki = 6.1 nM T05849 C73HPT 118727697 Ki = 1.2 nM T05849 C5C2RI 118727698 Ki = 3.7 nM T05849 C6Q9XZ 118727699 Ki = 30 nM T05849 C3ZNX5 135423404 Ki = 0.1072 nM T05849 CR79SC 135529065 Ki = 0.4266 nM T05849 C0OK8I 135610887 Ki = 0.1995 nM T05849 C8IP3M 136036821 Ki = 20.89 nM T05849 C6EOV2 136036823 Ki = 1.202 nM T05849 C15QJN 136046102 IC50 = 670 nM T05849 C8E7WR 136055865 IC50 = 0.266 nM T05849 CNE90O 136055866 IC50 = 56.4 nM T05849 C1UX8Y 136067266 IC50 = 80000 nM T05849 C0LPQ1 145978895 Ki = 7.93 nM T05849 CKL68T 145991328 Ki = 3.91 nM T05849 C48LWV 155512804 IC50 > 50000 nM T05849 CB89KA 155514270 EC50 > 1000 nM T05849 C9MB4S 155514432 IC50 = 128.82 nM T05849 CDK7N6 155515427 EC50 = 89.13 nM T05849 CL5KO6 155516160 IC50 = 25.8 nM T05849 C07LPH 155516677 IC50 = 0.2089 nM T05849 CBJH23 155517239 EC50 > 1000 nM T05849 CB1SI3 155517761 EC50 = 16.6 nM T05849 CBG5S4 155517868 EC50 = 0.8318 nM T05849 CU01ZN 155519400 IC50 = 25.4 nM T05849 CTV3M6 155521287 IC50 > 10000 nM T05849 C18CFP 155523323 IC50 = 200.5 nM T05849 CKC61A 155524181 EC50 = 0.4467 nM T05849 CH5AU4 155524770 IC50 = 3715.35 nM T05849 CAE58M 155526914 EC50 = 0.4169 nM T05849 C9HIR7 155530671 EC50 > 1000 nM T05849 C30VKS 155531277 EC50 = 5.754 nM T05849 CKL8Y2 155532425 EC50 = 0.631 nM T05849 CN0VP5 155532759 EC50 > 1000 nM T05849 C12IEY 155533399 EC50 = 0.2951 nM T05849 CVBR79 155533520 EC50 > 1000 nM T05849 CV5Z2P 155534566 IC50 = 1.7 nM T05849 CUBR54 155534993 IC50 = 15.4 nM T05849 CHV1D9 155535107 EC50 = 5.012 nM T05849 C09DZK 155535249 EC50 = 870.96 nM T05849 CNB7M5 155535579 EC50 = 1.549 nM T05849 C9MQD3 155536224 IC50 = 20.9 nM T05849 CKI3E1 155536333 EC50 > 1000 nM T05849 CO07KD 155537344 EC50 > 1000 nM T05849 C8QIH3 155539345 EC50 = 104.71 nM T05849 C2FBL5 155540394 EC50 = 25.7 nM T05849 CWP54F 155540415 EC50 = 0.3802 nM T05849 CMV82T 155540739 EC50 = 316.23 nM T05849 CB18RV 155542488 EC50 > 1000 nM T05849 CGN96I 155542545 EC50 > 1000 nM T05849 CY6E8B 155543163 EC50 = 173.78 nM T05849 CS5N7E 155543846 EC50 = 0.3236 nM T05849 C39DSM 155543995 EC50 > 1000 nM T05849 C7K4ZA 155544674 IC50 = 0.166 nM T05849 CLB1R7 155546692 EC50 = 0.4169 nM T05849 C7Z8OY 155547906 EC50 > 1000 nM T05849 CY9WQ0 155548021 IC50 = 15.6 nM T05849 C1PV3I 155548381 EC50 > 1000 nM T05849 CRW9Q8 155550030 IC50 = 18.8 nM T05849 C1GEA7 155550911 EC50 > 1000 nM T05849 CQ9S8X 155551968 EC50 > 1000 nM T05849 C1DG3Q 155552556 EC50 > 1000 nM T05849 C4QSR2 155553269 IC50 = 5370.32 nM T05849 C3K4NQ 155553502 EC50 = 0.3311 nM T05849 C51ZHW 155555065 EC50 = 131.83 nM T05849 C8V6RX 155555346 IC50 = 0.2884 nM T05849 CH5G6Q 155556375 IC50 = 8 nM T05849 CDF1E8 155557064 EC50 > 1000 nM T05849 CN68GS 155557285 EC50 = 0.3802 nM T05849 CO1N8R 155558199 EC50 = 0.4365 nM T05849 C0GE9L 155559320 IC50 = 0.09333 nM T05849 C2DFE4 155560670 EC50 = 1.862 nM T05849 CVKT21 155562102 IC50 > 50000 nM T05849 CLI24D 155562281 EC50 = 151.36 nM T05849 CFZ19O 155564367 EC50 = 0.3162 nM T05849 CFYB81 155564421 EC50 > 1000 nM T05849 CQ8G9E 155566319 EC50 = 123.03 nM T05849 CK98TD 155568312 EC50 = 2.692 nM T05849 CP23WI 44572148 Ki = 1 nM T05849 D00UKA 44272095 Ki = 54 nM T05849 D01ADK 11693641 Ki = 2.7 nM T05849 D01AQC 9811733 Ki = 15 nM T05849 D01FHK 3086453 IC50 = 0.2 nM T05849 D02ZML 5311148 IC50 = 1000 nM T05849 D03EHS 44272077 Ki = 313 nM T05849 D03EPA 11051303 Ki = 26 nM T05849 D03WGS 44408525 Ki = 1300 nM T05849 D03ZWL 132980 IC50 = 0.1 nM T05849 D05GQK 656755 IC50 = 13000 nM T05849 D05QBF 443375 Ki = 3.69 nM T05849 D05RRZ 10348659 IC50 = 251.19 nM T05849 D05XXE 446569 Ki = 10.4 nM T05849 D05YZC 59751 Ki = 169 nM T05849 D05ZUX 44207909 Ki >= 1000 nM T05849 D06BRA 11520765 EC50 = 323.59 nM T05849 D06DTT 193319 IC50 > 100000 nM T05849 D06NIP 11629355 IC50 = 0.2188 nM T05849 D07ICW 11556976 Ki = 1.3 nM T05849 D07LQQ 11564210 Ki = 15 nM T05849 D08QKT 11528076 Ki = 3.8 nM T05849 D09EMR 11136782 Ki = 1700 nM T05849 D09TNC 5311400 Ki = 0.28 nM T05849 D0A7RT 163781 EC50 = 1.5 nM T05849 D0E2OG 11614928 IC50 = 1096.48 nM T05849 D0EZ2W 45265542 IC50 = 700 nM T05849 D0F0MN 44272078 Ki = 334 nM T05849 D0F1XY 44408590 Ki > 10000 nM T05849 D0F8CV 5462471 EC50 = 2.66 nM T05849 D0H9AX 9935175 IC50 = 0.054 nM T05849 D0I8AF 9833444 EC50 = 0.05012 nM T05849 D0I9PH 16100409 Ki > 10000 nM T05849 D0J0CA 107704 IC50 = 150000 nM T05849 D0J7GJ 44408484 Ki = 9300 nM T05849 D0M1BJ 5282279 IC50 > 1000 nM T05849 D0M9GO 115208 Ki > 100000 nM T05849 D0N4QT 9953071 IC50 = 0.28 nM T05849 D0N6DN 44408524 Ki = 3800 nM T05849 D0O8HW 9872735 IC50 = 0.087 nM T05849 D0P9OL 44272056 Ki = 47.3 nM T05849 D0QP2S 44408526 Ki = 1500 nM T05849 D0R4GI 11040230 Ki = 1.6 nM T05849 D0S7SO 16100407 Ki = 71 nM T05849 D0T2RY 9948320 Ki >= 1000 nM T05849 D0TR0U 10942040 Ki = 1.1 nM T05849 D0U6OA 10909103 EC50 = 7.943 nM T05849 D0V0RB 11722088 IC50 = 2187.76 nM T05849 D0V9DY 16100410 Ki = 7700 nM T05849 D0X7LC 11061906 Ki = 1.3 nM T05849 D0Z4SS 44572147 Ki = 537.03 nM T01521 D00UVA 11556711 IC50 = 150 nM T01521 D01XNB 4594 IC50 = 4600 nM T01521 D06TNL 3278 IC50 = 25000 nM T01521 D0G3DL 135398735 IC50 = 75000 nM T01521 D0QG8F 6 IC50 = 900000 nM T01521 C05CMQ 20353 IC50 = 4000 nM T01521 CPW9G5 65126 IC50 = 62000 nM T01521 CZ5G2B 94493 IC50 = 2000 nM T01521 CX4VQ7 185710 IC50 < 400 nM T01521 CH37YQ 3816252 IC50 = 160 nM T01521 CQ4B9M 3850682 IC50 = 120 nM T01521 CDO03H 3860347 IC50 = 21 nM T01521 CU28PK 4257368 IC50 = 28 nM T01521 CI57VC 4380267 IC50 = 54 nM T01521 CYH24L 9888140 IC50 = 250 nM T01521 CXD85M 11644907 IC50 = 1600 nM T01521 CG5Y0L 12643450 IC50 = 470 nM T01521 CC6JA9 16226974 IC50 > 10000 nM T01521 CX7Y2N 23668196 IC50 = 1020000 nM T01521 CLT8X7 43405493 IC50 = 1010 nM T01521 C30KAW 43405519 IC50 = 4490 nM T01521 CYJ0X3 43405535 IC50 = 880 nM T01521 C64TZL 43406232 IC50 = 3140 nM T01521 CMD17V 43415488 IC50 > 10000 nM T01521 CNQ85W 43616381 IC50 > 10000 nM T01521 C3HC9U 43616626 IC50 = 810 nM T01521 CNQ8O6 43616650 IC50 = 220 nM T01521 CB2Y9J 53364469 IC50 = 21 nM T01521 CM82RO 54867190 IC50 > 10000 nM T01521 C1DJU5 60948880 IC50 > 10000 nM T01521 C1DTS2 71466696 IC50 = 13000 nM T01521 C92KHU 76900024 IC50 = 40 nM T01521 C51FKG 118553182 IC50 = 350 nM T01521 CR8OC3 122144039 IC50 > 10000 nM T01521 C80JPQ 132040441 IC50 = 400 nM T01521 CUCG67 138857439 IC50 = 80 nM T01521 C3K9VW 138857440 IC50 = 70 nM T01521 CG8X7A 139226240 IC50 = 170 nM T01521 CBU65E 146025594 IC50 = 250 nM T01521 CTH7I3 155511072 IC50 = 150 nM T01521 CE4WL8 155511172 IC50 = 3200 nM T01521 CN1G5W 155512763 IC50 = 110 nM T01521 C31LNR 155514182 IC50 = 580 nM T01521 CH5K3B 155515269 IC50 > 100000 nM T01521 CYL95S 155515371 IC50 = 1580 nM T01521 CMFI31 155515426 IC50 = 340 nM T01521 CN1OK4 155516600 IC50 = 25 nM T01521 CIKW40 155516831 IC50 = 80 nM T01521 CG9A5P 155517058 IC50 = 740 nM T01521 CNGI52 155517253 IC50 = 30 nM T01521 C80FZB 155517269 IC50 > 10000 nM T01521 CBCA63 155517428 IC50 = 370 nM T01521 CO7GK3 155517915 IC50 = 3110 nM T01521 C56NVF 155520859 IC50 = 160 nM T01521 CS7L9X 155522104 IC50 > 100000 nM T01521 CD6CO1 155523627 IC50 = 51 nM T01521 C3VGS7 155524556 IC50 = 230 nM T01521 CRO65L 155526238 IC50 = 600 nM T01521 CB5S8Q 155526467 IC50 = 270 nM T01521 COKJ87 155527110 IC50 = 60 nM T01521 CHO80A 155529864 IC50 = 5.6 nM T01521 CC5P9U 155531289 IC50 = 180 nM T01521 CI20PV 155536137 IC50 = 1220 nM T01521 CV3I6D 155536315 IC50 = 300 nM T01521 C05BFR 155536500 IC50 > 10000 nM T01521 CKT62R 155537169 IC50 = 1030 nM T01521 C2ULE7 155537449 IC50 = 150 nM T01521 C29DSR 155538240 IC50 = 710 nM T01521 CCQ7P9 155539037 IC50 = 0.32 nM T01521 CL05KP 155539569 IC50 > 10000 nM T01521 CJ0E2O 155539725 IC50 > 10000 nM T01521 CK3ZI8 155542111 IC50 = 200 nM T01521 CGN4L1 155543255 IC50 = 190 nM T01521 CZA39M 155545567 IC50 = 30 nM T01521 C7Q5UO 155546251 IC50 = 860 nM T01521 CA0VC9 155551747 IC50 > 100000 nM T01521 CHB4D2 155552757 IC50 = 210 nM T01521 C31DBM 155553666 IC50 > 10000 nM T01521 CR8NI7 155554345 IC50 = 360 nM T01521 CGO7D0 155554862 IC50 = 720 nM T01521 CA70KB 155556475 IC50 = 800 nM T01521 C62DEC 155556999 IC50 = 570 nM T01521 CI4BR7 155557257 IC50 > 10000 nM T01521 CR65JL 155559750 IC50 > 100000 nM T01521 CCX81U 155560442 IC50 = 40 nM T01521 C0U6TX 155561402 IC50 = 700 nM T01521 CNA8R4 155563174 IC50 = 530 nM T01521 CV4LZ3 155563229 IC50 > 100000 nM T01521 CE8Y4W 155564541 IC50 > 1000000 nM T01521 C5D8AS 155565457 IC50 = 1200 nM T01521 CR42VB 155566134 IC50 = 2040 nM T01521 CN03FV 155566179 IC50 = 1290 nM T01521 C7PEH6 155567328 IC50 = 130 nM T01521 CLWA82 155569650 IC50 = 0.22 nM T39486 D05ADP 160355 IC50 = 1700 nM T39486 D06DMQ 59472121 Ki = 26 nM T39486 D0E3TC 44259 IC50 = 248 nM T39486 D03BNU 59604787 IC50 > 10000 nM T39486 D00OWF 5280953 IC50 = 900 nM T39486 D0NS6I 10037501 IC50 = 1500 nM T39486 D0Q3VZ 135398522 IC50 = 35 nM T39486 D0WX0K 71680628 IC50 = 530 nM T39486 C1B9ZO 68094 IC50 = 1500 nM T39486 CVMO57 95875 IC50 > 10000 nM T39486 CN6AY0 491467 IC50 = 6300 nM T39486 C3D1HC 762415 IC50 > 10000 nM T39486 CFA92X 1237489 IC50 > 10000 nM T39486 CD1A9T 1241605 IC50 > 10000 nM T39486 CO6KI2 5930298 IC50 = 990 nM T39486 CLN2G8 6475560 IC50 = 1100 nM T39486 CACS26 11561968 Ki > 2000 nM T39486 CP04JC 11666231 IC50 = 60 nM T39486 CU0E8O 11690457 Ki > 2000 nM T39486 CPI54D 11953235 IC50 = 166 nM T39486 C38FDZ 16760660 IC50 = 950 nM T39486 CMW42V 19079253 IC50 = 9200 nM T39486 CY8L7E 24896769 IC50 > 10000 nM T39486 CQ0ZI7 45141513 IC50 = 11000 nM T39486 CE4SU5 47298428 IC50 = 1000 nM T39486 C1XP7K 53308973 IC50 = 5100 nM T39486 CBPV19 53308974 IC50 = 6500 nM T39486 C58TBY 53308976 IC50 = 1100 nM T39486 C2CH7R 53309118 IC50 = 510 nM T39486 CDV5X6 53309119 IC50 = 100 nM T39486 C2QW5D 53309120 IC50 = 120 nM T39486 C65OUB 54575585 IC50 > 10000 nM T39486 CUA4K6 54575586 IC50 > 10000 nM T39486 CY46FV 54575645 IC50 > 10000 nM T39486 C3CI0P 54575646 IC50 > 10000 nM T39486 C2CS9V 54575647 IC50 > 10000 nM T39486 CKMU37 54575648 IC50 > 10000 nM T39486 CU02GP 54575649 IC50 > 10000 nM T39486 CI38EN 54575650 IC50 > 10000 nM T39486 C4A5PV 54575651 IC50 = 4900 nM T39486 C39YTB 54575652 IC50 = 7000 nM T39486 C7XEO8 54575715 IC50 = 8000 nM T39486 CG4TF1 54575716 IC50 > 10000 nM T39486 CNCR40 54575717 IC50 > 10000 nM T39486 CKU8H1 54575718 IC50 > 10000 nM T39486 CKFP41 54575720 IC50 > 10000 nM T39486 C4E3PA 54575721 IC50 = 8500 nM T39486 C9SY1C 54575783 IC50 = 4800 nM T39486 CQ1KA8 54613080 IC50 = 15000 nM T39486 CFB2R8 56676630 IC50 = 460 nM T39486 CDK93W 56946894 IC50 = 40 nM T39486 CR3I5F 57418686 IC50 = 1300 nM T39486 CF6K1Y 58857683 IC50 = 7000 nM T39486 C56MAG 59379853 IC50 = 480 nM T39486 CV63UL 67240318 IC50 > 10000 nM T39486 CBY80T 72716071 IC50 = 190000 nM T39486 C4BV9L 73426232 IC50 > 1000 nM T39486 CVD5U4 76314850 IC50 = 1400 nM T39486 C0GYK1 86765296 IC50 = 1700 nM T39486 C4BKA6 89429109 IC50 = 8600 nM T39486 C2FOK4 89494280 IC50 = 820 nM T39486 CE5L8V 90388565 IC50 = 610 nM T39486 CWE9I2 91664021 IC50 > 10000 nM T39486 CW58AE 91664022 IC50 = 220 nM T39486 CB25UZ 91664023 IC50 = 130 nM T39486 CO83PN 122181013 IC50 = 40 nM T39486 C69ULZ 122181014 IC50 = 16 nM T39486 CIG8Y1 122181016 IC50 = 8000 nM T39486 CRJS41 122181017 IC50 = 33 nM T39486 CVB03H 122181018 IC50 = 23 nM T39486 C6SJ3X 122181019 IC50 > 10000 nM T39486 C7L5PG 122181021 IC50 > 10000 nM T39486 C58CJI 122181022 IC50 > 10000 nM T39486 CC2G8N 122181024 IC50 = 79 nM T39486 CV5BQ9 122181097 IC50 > 10000 nM T39486 C5KB1C 122184057 IC50 = 40 nM T39486 CVBF01 127030212 IC50 = 430 nM T39486 CI93ZA 127030213 IC50 = 2040 nM T39486 C8LQV4 127030516 IC50 > 10000 nM T39486 CS12RU 127031435 IC50 = 200 nM T39486 CZXP62 127031750 IC50 > 10000 nM T39486 C3E5YO 127032014 IC50 = 60 nM T39486 C2ZD8S 127032024 IC50 = 1500 nM T39486 CXWY73 127032324 IC50 = 820 nM T39486 C2LWZ1 129318964 IC50 > 10000 nM T39486 CM8DK3 134813913 IC50 = 120 nM T39486 C9QI4V 135423788 IC50 > 10000 nM T39486 CEVL69 135423792 IC50 = 1300 nM T39486 CTAC32 135423796 IC50 > 10000 nM T39486 CBU0J4 135604653 IC50 > 10000 nM T39486 C1KP2E 135860183 IC50 = 710 nM T39486 CGX7J5 135885107 IC50 = 1600 nM T39486 CR1P5M 136025848 IC50 = 610 nM T39486 CG39ZH 136025849 IC50 = 2000 nM T39486 C85XKB 136025991 IC50 = 2200 nM T39486 CC4UG2 136025994 IC50 = 40 nM T39486 C63KRL 136026134 IC50 > 10000 nM T39486 CKL49A 136026136 IC50 = 120 nM T39486 C1HV2M 136026137 IC50 = 47 nM T39486 CTX08I 136026138 IC50 = 550 nM T39486 CBO76R 136026139 IC50 = 560 nM T39486 C8QU9L 136026140 IC50 = 470 nM T39486 C7OKA9 136033523 IC50 = 210 nM T39486 CV0U7E 136033524 IC50 = 620 nM T39486 CHQO83 136033525 IC50 = 340 nM T39486 CO34IK 136033527 IC50 = 6000 nM T39486 CQS9R7 136033528 IC50 = 770 nM T39486 CD1A7S 136033529 IC50 = 560 nM T39486 C6VH4F 136033539 IC50 > 10000 nM T39486 C4H9ZD 136033543 IC50 > 10000 nM T39486 CC54MD 136033544 IC50 = 160 nM T39486 C2AO3G 136033545 IC50 = 61 nM T39486 CJ98EN 136033546 IC50 = 60 nM T39486 C3I7UD 136033547 IC50 = 80 nM T39486 CVFW17 136033548 IC50 = 110 nM T39486 CSV8T4 136068690 IC50 = 2100 nM T39486 CCVU40 136086892 IC50 = 640 nM T39486 CHR1T4 136086893 IC50 = 530 nM T39486 CM84LZ 136086894 IC50 = 10000 nM T39486 C13DGL 136086895 IC50 = 3300 nM T39486 CH0Q2Z 136234577 IC50 = 150 nM T39486 CV6F4N 136234578 IC50 = 130 nM T39486 C2G3JY 136234579 IC50 > 10000 nM T39486 CJ2F7R 136238979 IC50 > 10000 nM T39486 CT3KB7 136238980 IC50 > 10000 nM T39486 C8JGC6 136238981 IC50 > 10000 nM T39486 CJDO36 136238982 IC50 > 10000 nM T39486 CY6M7W 136239000 IC50 > 10000 nM T39486 CF1V6K 136239001 IC50 = 1100 nM T39486 C8G7OB 136239002 IC50 > 10000 nM T39486 CH17EC 136239003 IC50 > 10000 nM T39486 C3IV7E 136239004 IC50 = 1300 nM T39486 C0PQ5H 136239005 IC50 > 10000 nM T39486 CZ76FY 136239019 IC50 > 10000 nM T39486 CFUZ87 136240995 IC50 = 1800 nM T39486 CO17AY 136252249 IC50 > 10000 nM T39486 CCAZ26 137631656 IC50 = 390 nM T39486 C3QAV9 137631819 IC50 = 1800 nM T39486 CI43OC 137632412 IC50 = 644 nM T39486 CG8Y0U 137633419 IC50 = 21000 nM T39486 CH4PN9 137633814 IC50 = 476 nM T39486 CS9TU2 137633985 IC50 = 1200 nM T39486 C83UKG 137634382 IC50 = 210 nM T39486 CNT7S3 137634818 IC50 > 10000 nM T39486 CCP7X5 137635304 IC50 = 2500 nM T39486 C1AK8X 137635556 IC50 = 3200 nM T39486 CV7OF5 137635713 IC50 = 10000 nM T39486 C5QWE1 137635926 IC50 = 43 nM T39486 CKZF46 137638065 IC50 > 10000 nM T39486 CRV1E4 137638175 IC50 > 1000 nM T39486 CCX37E 137638472 IC50 = 82 nM T39486 CPO87L 137638509 IC50 = 48 nM T39486 C1UI5N 137638944 IC50 = 2500 nM T39486 CH4RP3 137639514 IC50 = 440 nM T39486 CX3MQ1 137639546 IC50 = 500 nM T39486 CH3S8N 137640038 IC50 = 170 nM T39486 CXM4G7 137640811 IC50 = 190 nM T39486 CF83TG 137640934 IC50 = 110 nM T39486 CRSQ71 137641785 IC50 = 408 nM T39486 CWVE69 137643514 IC50 = 440 nM T39486 CYA1F7 137643721 IC50 = 120 nM T39486 C2AG3W 137643887 IC50 = 19000 nM T39486 C4DS3I 137643955 IC50 = 1900 nM T39486 C75MLQ 137643957 IC50 = 724 nM T39486 CWIP72 137644498 IC50 = 380 nM T39486 CZ4U0W 137644802 IC50 = 180 nM T39486 CPJ42V 137644974 IC50 > 10000 nM T39486 C8VTQ9 137645650 IC50 = 400 nM T39486 C7ZOV3 137645947 IC50 > 10000 nM T39486 CL5NX9 137646497 IC50 = 1200 nM T39486 CJ5O2Q 137646673 IC50 = 3000 nM T39486 CK6S5T 137646758 IC50 > 1000 nM T39486 COU37W 137647335 IC50 = 380 nM T39486 CMI2H3 137647526 IC50 = 571 nM T39486 C7O2AW 137647969 IC50 > 10000 nM T39486 CNW13G 137648784 IC50 > 1000 nM T39486 CGK5P2 137649037 IC50 > 1000 nM T39486 C5OJH2 137649318 IC50 = 730 nM T39486 C9IO5F 137649821 IC50 = 536 nM T39486 C9QNG8 137650421 IC50 = 8200 nM T39486 CWG94C 137650926 IC50 = 7200 nM T39486 C8MKN0 137651314 IC50 = 320 nM T39486 CKL0P4 137651538 IC50 = 3900 nM T39486 CJ14XO 137651668 IC50 = 1400 nM T39486 CH6L2T 137652047 IC50 = 1600 nM T39486 C2B5CY 137652970 IC50 = 1600 nM T39486 C48DVU 137653000 IC50 = 120 nM T39486 C01URE 137653446 IC50 > 10000 nM T39486 CDX83M 137654129 IC50 = 567 nM T39486 C47FBV 137654225 IC50 = 3100 nM T39486 CX7V6P 137654671 IC50 > 1000 nM T39486 C7IU4J 137655848 IC50 = 63 nM T39486 CQEJ60 137656868 IC50 = 40 nM T39486 C3Y2CR 137657691 IC50 = 416 nM T39486 CA10CX 137657812 IC50 = 847 nM T39486 C39SEV 137658150 IC50 = 780 nM T39486 CX8YL9 137658187 IC50 = 50 nM T39486 CX4M8T 137658722 IC50 > 1000 nM T39486 CA2PY1 137658970 IC50 = 600 nM T39486 CJ1TB2 137659239 IC50 = 4500 nM T39486 C3U2OB 137659350 IC50 = 600 nM T39486 C7MI2G 137661183 IC50 = 6300 nM T39486 CIX41F 137661315 IC50 = 7100 nM T39486 CD0FV8 137661355 IC50 = 1200 nM T39486 CO1S8D 145986658 IC50 = 490 nM T39486 C7SOT2 145987707 IC50 = 5000 nM T39486 C2MD1Q 155513187 IC50 > 10000 nM T39486 D08NQM 5289247 IC50 = 100 nM T01211 CGAX04 6436223 IC50 = 100 nM T01211 CBJK75 9848597 IC50 > 10000 nM T01211 C0BF6T 10649263 IC50 > 10000 nM T01211 C1TV6X 23238906 IC50 > 10000 nM T01211 CGEU75 44286299 IC50 = 1900 nM T01211 CW3RE5 44299337 IC50 > 10000 nM T01211 CM6BX4 44299391 IC50 > 10000 nM T67416 CR6HO1 8593 IC50 > 100000 nM T67416 C7V6ZI 26587 IC50 > 100000 nM T67416 C5KLH7 230595 IC50 > 100000 nM T67416 C14JKX 487529 Ki = 5.1 nM T67416 C9QJ6X 625773 IC50 > 100000 nM T67416 C80TDH 676325 IC50 > 100000 nM T67416 C74ZEV 680333 IC50 > 100000 nM T67416 COE1U4 695258 IC50 > 100000 nM T67416 C7WEV5 697640 IC50 > 100000 nM T67416 CD41EI 997453 IC50 > 100000 nM T67416 C7BZF2 1016084 IC50 > 100000 nM T67416 CDA1B6 1038445 IC50 > 20000 nM T67416 C1Q3XA 1223599 IC50 > 20000 nM T67416 CVN4U7 4038525 IC50 > 100000 nM T67416 CTN59F 5275522 IC50 > 100000 nM T67416 C4T0GK 5275524 IC50 = 95000 nM T67416 CYHV40 5275525 IC50 = 80000 nM T67416 CT9W3I 5275526 IC50 = 35000 nM T67416 C9D8GK 5275527 IC50 > 100000 nM T67416 C45HGL 5275528 IC50 > 20000 nM T67416 CJF1D4 5275530 IC50 > 100000 nM T67416 CPR46U 5275531 IC50 = 56000 nM T67416 C7FG5P 5275532 IC50 = 70000 nM T67416 C59IES 5275533 IC50 = 60000 nM T67416 C0Y9UV 5275535 IC50 > 100000 nM T67416 CBD21C 5275536 IC50 > 100000 nM T67416 CDS05Z 5275537 IC50 > 100000 nM T67416 C6E8XB 5275538 IC50 > 100000 nM T67416 CB4DM3 44367066 IC50 > 100000 nM T67416 CRBW52 44367229 IC50 > 100000 nM T67416 CX4JU3 44367351 IC50 > 100000 nM T18299 D0W8SJ 4199 IC50 > 100000 nM T18299 D0E3TC 44259 IC50 = 2 nM T18299 D0I6VU 176167 IC50 = 10000 nM T18299 D0W3LI 153999 IC50 = 6200 nM T18299 D0Z1DH 10029385 IC50 > 20000 nM T18299 C8NW5J 3815 IC50 = 184 nM T18299 C4MNG8 445840 IC50 > 10000 nM T18299 CB9F1O 447961 Ki > 1000 nM T18299 C4VTS3 5327723 IC50 = 25 nM T18299 CZ3LK2 5330387 IC50 > 10000 nM T18299 CRU94N 5330388 IC50 > 10000 nM T18299 CDB68F 5330389 IC50 > 10000 nM T18299 C7CX0H 5330390 IC50 > 10000 nM T18299 C8E0XS 5330391 IC50 > 10000 nM T18299 CW1VX9 5330392 IC50 > 10000 nM T18299 C67DRP 5330708 IC50 > 2000 nM T18299 CND03V 5330710 IC50 = 174 nM T18299 C74ZYC 5330764 IC50 = 6120 nM T18299 C2EQO4 5330765 IC50 > 20000 nM T18299 CE9F5H 5330766 IC50 = 527 nM T18299 CT65PW 5330767 IC50 = 1170 nM T18299 CI07AT 5330768 IC50 = 3050 nM T18299 C5EX0R 5330769 IC50 = 3130 nM T18299 CIV65Z 5330770 IC50 = 11600 nM T18299 CV69TO 5330771 IC50 = 732 nM T18299 C81SBW 5330772 IC50 > 20000 nM T18299 C1Z6LK 5330773 IC50 > 20000 nM T18299 C65YDC 5330774 IC50 = 81 nM T18299 CTRP80 5330775 IC50 = 25 nM T18299 C6CI5V 5330776 IC50 = 301 nM T18299 CQCL86 5330777 IC50 = 46 nM T18299 CDTH41 5330778 IC50 = 90 nM T18299 C7R6HB 5330779 IC50 = 62 nM T18299 CD7UK4 5330780 IC50 = 95 nM T18299 CP18GL 5330781 IC50 = 177 nM T18299 CSB6J8 5330782 IC50 = 403 nM T18299 CAT2Z5 5330783 IC50 = 49 nM T18299 CR6D1C 5330784 IC50 = 382 nM T18299 CRB01P 5330785 IC50 = 266 nM T18299 C8UI2M 5330786 IC50 = 516 nM T18299 C1F7DP 5330787 IC50 = 174 nM T18299 C31FHN 5330788 IC50 = 216 nM T18299 CU5W8P 5330791 IC50 = 914 nM T18299 C5O0CF 5330792 IC50 > 2000 nM T18299 CA3MY8 5330793 IC50 = 236 nM T18299 C3V6BO 5330794 IC50 > 2000 nM T18299 C0G3BP 5330795 IC50 = 58 nM T18299 CDGW17 5330796 IC50 < 1250 nM T18299 CL2G0Z 5330798 IC50 = 11100 nM T18299 CIHU71 5330799 IC50 = 92 nM T18299 CE68TK 5330801 IC50 = 82 nM T18299 CF01JS 5330804 IC50 = 10500 nM T18299 CL47HK 9795307 IC50 = 760000 nM T18299 C8J1OL 9826373 IC50 = 25000 nM T18299 C20NKA 9889351 IC50 = 2000 nM T18299 CQD2W7 9935079 IC50 > 10000 nM T18299 CV34AB 9958125 IC50 > 40000 nM T18299 C70FVS 10102940 IC50 > 200000 nM T18299 CZJI60 10141037 IC50 > 10000 nM T18299 C94WRY 10143231 IC50 > 10000 nM T18299 C5P8JC 10206423 IC50 > 10000 nM T18299 CGOT91 10207821 IC50 = 780 nM T18299 CPVZ80 10329065 IC50 > 200000 nM T18299 C18ATD 10369873 IC50 > 100000 nM T18299 CO8FU3 10534425 IC50 > 200000 nM T18299 C8EI5N 10534451 IC50 > 200000 nM T18299 C5MZ0F 10534468 IC50 = 16200 nM T18299 CHUM60 10558336 IC50 > 200000 nM T18299 C8EZM4 10558364 IC50 > 200000 nM T18299 CW0O2T 10582255 IC50 > 200000 nM T18299 CW0ER3 10606421 IC50 > 200000 nM T18299 C02DWP 10654010 IC50 > 200000 nM T18299 C57BUS 10677930 IC50 = 132000 nM T18299 C2F4RJ 10677940 IC50 > 200000 nM T18299 CK8P6M 10701564 IC50 > 200000 nM T18299 CZ7NC2 10701654 IC50 = 26700 nM T18299 CB82QD 10725077 IC50 > 200000 nM T18299 CRE4Y9 10772744 IC50 > 200000 nM T18299 CFB2P1 10820190 IC50 > 200000 nM T18299 C1L4ZC 10940039 IC50 = 59000 nM T18299 C2W5RC 11235063 IC50 > 50000 nM T18299 C30PKR 11248978 IC50 > 20000 nM T18299 CSXY78 11294864 IC50 > 20000 nM T18299 CPU9I3 11316975 IC50 = 2500 nM T18299 CQ8I4H 11328863 IC50 > 20000 nM T18299 C8DNQ2 11453012 IC50 = 2000 nM T18299 CK34LS 11632737 IC50 > 50000 nM T18299 CCX53Q 11729563 IC50 = 3000 nM T18299 C8AH1I 17758019 IC50 > 100000 nM T18299 C1GKL6 17758020 IC50 = 5600 nM T18299 CIE58R 17758239 IC50 > 40000 nM T18299 CO6LR5 17758240 IC50 > 40000 nM T18299 CWH37T 17758574 IC50 > 40000 nM T18299 C57NRL 17759787 IC50 > 40000 nM T18299 CVR9K4 22907281 IC50 = 7500 nM T18299 C0HRM6 22911602 IC50 = 7000 nM T18299 C9L4SQ 24955953 IC50 > 100000 nM T18299 CG9YQ3 44267896 IC50 = 36 nM T18299 CG5XC9 44267897 IC50 = 1200 nM T18299 C0ZX6Y 44267898 IC50 = 1000 nM T18299 CH28JU 44343747 IC50 > 100000 nM T18299 C6MK9J 44383010 IC50 > 200000 nM T18299 CB04FM 44383011 IC50 > 200000 nM T18299 C31SXF 44383381 IC50 = 57400 nM T18299 C3GD4Q 44384042 IC50 > 200000 nM T18299 CT76PJ 44384241 IC50 > 200000 nM T18299 CE32KB 44384242 IC50 > 200000 nM T18299 C51KYU 44384243 IC50 > 200000 nM T18299 CSBC59 44396134 IC50 > 20000 nM T18299 CW3BP8 44398371 IC50 > 100000 nM T18299 C9S5DT 56668086 IC50 > 200000 nM T18299 CCVA54 73356021 IC50 = 32 nM T18299 D03MUZ 17759555 IC50 > 40000 nM T18299 D04NGS 5330790 IC50 > 100000 nM T18299 D07OCA 5330812 IC50 = 8900 nM T18299 D0D5HQ 5330797 IC50 = 12400 nM T84040 D04CSZ 1254 EC50 = 28400 nM T84040 D05FTJ 4044 EC50 = 16000 nM T84040 D06GIP 6989 EC50 = 6000 nM T84040 D0B2WJ 3371 EC50 = 6918.31 nM T84040 D0BQ8Y 5971 EC50 = 398 nM T84040 D0E6OC 5282230 IC50 = 125892.54 nM T84040 D0L7FM 4911 EC50 = 4200000 nM T84040 D0T8GD 89594 EC50 = 2000 nM T84040 D0TG1H 3033 EC50 = 56000 nM T84040 D0X5SD 3117 EC50 = 3000 nM T84040 D00KTV 5469318 EC50 = 800 nM T84040 D07AOL 16741 EC50 = 370 nM T84040 D0C0NH 3806 EC50 = 1700 nM T84040 D0CO6D 71144018 IC50 > 40000 nM T84040 D0U3EP 445154 IC50 = 750 nM T84040 D0DK4I 4534 EC50 = 4900 nM T84040 D0O4QB 3314 EC50 = 168000 nM T84040 CT3IS2 2346 EC50 = 250 nM T84040 CHNF82 7748 EC50 = 39 nM T84040 CU3LG2 9213 EC50 = 0.3 nM T84040 CC9O7U 11443 EC50 = 10000 nM T84040 C49FZU 11617 EC50 = 254000 nM T84040 CY7J1X 16315 EC50 = 490 nM T84040 CJS35X 16590 EC50 = 7550 nM T84040 C9V3ZD 16666 EC50 = 96000 nM T84040 CD1J2P 22044 EC50 = 10 nM T84040 CTDN51 62351 EC50 = 450 nM T84040 CX08SN 68381 EC50 = 19700 nM T84040 C94RLC 68960 EC50 = 690 nM T84040 C2NM4A 72503 EC50 = 59 nM T84040 C76SDU 75263 EC50 = 530 nM T84040 CZB4P2 76922 EC50 = 360 nM T84040 C7UD3V 78151 EC50 = 680 nM T84040 CK3D8C 78160 EC50 = 420 nM T84040 CK42MC 87436 EC50 = 540 nM T84040 CX3KQ1 91457 EC50 = 33000 nM T84040 C07UZO 123411 EC50 = 18400 nM T84040 CKU84Y 159055 IC50 = 400000 nM T84040 CTEY14 160611 EC50 = 20000 nM T84040 C8JOI2 165224 EC50 = 580 nM T84040 C6H0VW 184852 EC50 = 1040 nM T84040 C1UI5X 206037 EC50 = 500 nM T84040 CBT7O2 413295 EC50 = 1580 nM T84040 CGF6W2 642376 IC50 = 23000 nM T84040 CZTS52 693136 EC50 = 30000 nM T84040 C7G3WY 838375 IC50 > 10000 nM T84040 C41GCS 1146273 IC50 < 1000 nM T84040 C6AHJ5 1164343 IC50 < 1000 nM T84040 CR37XU 1245920 IC50 = 12100 nM T84040 CJ1U8Q 2302297 EC50 = 9 nM T84040 CH0D8L 2400427 EC50 = 49000 nM T84040 CRHE73 2463055 EC50 = 125892.54 nM T84040 C8BJ3A 3093506 IC50 = 1700 nM T84040 C64WRH 3237127 IC50 > 10000 nM T84040 CJ89FI 3821210 IC50 = 1400 nM T84040 CAQL74 4809029 IC50 > 16700 nM T84040 CL9Z4S 5029397 IC50 < 1000 nM T84040 CA9Q6P 5319022 EC50 = 44000 nM T84040 CWEQ47 5353623 EC50 = 90000 nM T84040 CU7MX6 5375953 IC50 = 1700 nM T84040 CJ3F1M 5384164 IC50 > 10000 nM T84040 C25YUO 5458190 EC50 = 9000 nM T84040 CX56UR 5704879 IC50 = 1700 nM T84040 CR68NF 5996309 EC50 = 199526.23 nM T84040 CS6E7A 6013922 EC50 = 75000 nM T84040 C3LFG7 6443019 IC50 = 43000 nM T84040 C12KZB 6552009 IC50 = 300000 nM T84040 C8QH2T 6977766 IC50 = 110 nM T84040 CHE70V 9838722 EC50 > 30000 nM T84040 C43NXF 9859693 EC50 = 9800 nM T84040 CS6FN7 9883254 IC50 = 550 nM T84040 CP92WJ 9884140 EC50 = 26915.35 nM T84040 C0GC4S 10027372 EC50 > 25000 nM T84040 CG4IY8 10059651 EC50 > 30000 nM T84040 CB34HN 10084135 EC50 = 6600 nM T84040 C75BPC 10115694 IC50 = 1460 nM T84040 CE7H8R 10125146 EC50 = 610 nM T84040 CMWN62 10137111 IC50 = 2230 nM T84040 CC6YK5 10138119 IC50 = 2230 nM T84040 C7JPL9 10158171 IC50 = 1880 nM T84040 CKI74T 10158248 IC50 = 1170 nM T84040 CHY9Z6 10180373 IC50 = 1370 nM T84040 C4SCL3 10183856 IC50 = 1740 nM T84040 C12OFQ 10201365 IC50 = 1570 nM T84040 CQV50C 10206095 IC50 = 680 nM T84040 CV81KY 10294753 IC50 = 3490 nM T84040 CW9VR1 11508468 EC50 = 11481.54 nM T84040 CH3F1I 11514966 EC50 = 42000 nM T84040 CQEK72 11515763 EC50 > 25000 nM T84040 CWG5M0 11536089 EC50 > 30000 nM T84040 CH5FP7 11551205 EC50 = 10000 nM T84040 C6LS3P 11571834 EC50 = 1050 nM T84040 CDZX61 11658617 EC50 = 83600 nM T84040 CB5W3T 11666329 EC50 = 149000 nM T84040 CV3RW9 12110672 EC50 = 78000 nM T84040 C2R0VQ 12286507 EC50 = 14 nM T84040 CE38OM 12444907 EC50 = 42000 nM T84040 CLR16B 15240186 IC50 > 30000 nM T84040 COL7M1 17421069 IC50 = 685 nM T84040 CTP2C3 18690881 EC50 = 0.15 nM T84040 C4MX5B 21468844 IC50 = 1290 nM T84040 CD6H7C 21598349 EC50 = 8000 nM T84040 CCG43N 22296670 EC50 = 32000 nM T84040 C8U7MH 26642769 IC50 = 10000 nM T84040 CLY1V2 27007581 IC50 > 8330 nM T84040 C9F6ZH 27010025 IC50 = 802 nM T84040 CTLK58 27017804 IC50 > 16700 nM T84040 C2RT9P 31538897 IC50 > 32000 nM T84040 C9FBE2 32622575 IC50 < 1000 nM T84040 CCA3M2 32682004 IC50 = 6600 nM T84040 C1E9SH 42609882 EC50 = 0.05 nM T84040 CZN60W 42635157 EC50 = 100 nM T84040 CAV28S 42635158 EC50 = 0.1 nM T84040 C3NC4B 42635159 EC50 = 245 nM T84040 CK3C9V 42635160 EC50 = 40 nM T84040 CC21XP 42635161 EC50 = 2.5 nM T84040 C1QNC4 42635336 EC50 = 6 nM T84040 CCAM65 42635337 EC50 = 6.2 nM T84040 CS1GF3 42635340 EC50 = 933 nM T84040 CH1VO9 42635341 EC50 = 0.07586 nM T84040 CZL26K 42635342 EC50 = 31 nM T84040 CHUX57 42635520 EC50 = 31 nM T84040 CA9Y8K 42635521 EC50 = 19 nM T84040 CUD9G4 42635522 EC50 = 0.11 nM T84040 CFP2S3 42635523 EC50 = 0.1175 nM T84040 CY3CT2 42641861 IC50 = 67 nM T84040 C92JAX 44224229 IC50 < 250 nM T84040 C63ZPV 44232532 EC50 = 830 nM T84040 CS4KX3 44241798 IC50 = 500 nM T84040 CDB9N1 44241929 IC50 = 250 nM T84040 C9X6JZ 44241930 IC50 = 250 nM T84040 C8W7TK 44241932 IC50 = 250 nM T84040 C1N5XF 44242814 IC50 = 500 nM T84040 C2XM9I 44448710 EC50 = 134000 nM T84040 CC6F7A 44448729 EC50 = 100 nM T84040 C4IT7J 44464276 EC50 = 4400 nM T84040 C75LAU 44464277 EC50 = 4450 nM T84040 CR7D0J 44464279 EC50 = 3000 nM T84040 CRE73L 44464525 EC50 = 510 nM T84040 CYPZ24 44464526 EC50 = 610 nM T84040 CK4Q1X 44464527 EC50 = 1160 nM T84040 C2EVO5 44464773 EC50 = 1290 nM T84040 C31TOX 44480618 IC50 < 1000 nM T84040 CN6WU1 44480883 IC50 < 1000 nM T84040 CXQ08U 44540055 IC50 = 30 nM T84040 CC31AH 44566752 EC50 = 30000 nM T84040 C6GM7Q 45257938 IC50 = 16100 nM T84040 C4WS8T 45375957 EC50 > 25000 nM T84040 CBI2C3 46879825 EC50 = 1600 nM T84040 CP4T7X 46879826 EC50 = 1800 nM T84040 CAQ5R4 46879827 EC50 = 3100 nM T84040 C3DZ7T 46879828 EC50 = 2000 nM T84040 CE35RZ 46879878 EC50 = 600 nM T84040 CVI20B 46879879 EC50 = 1000 nM T84040 C7YUV0 46879880 EC50 > 25000 nM T84040 CQ7BG8 46879881 EC50 > 25000 nM T84040 C17SUC 46879882 EC50 > 25000 nM T84040 C3KJD7 46879962 EC50 > 25000 nM T84040 CBK1A2 46879963 EC50 > 25000 nM T84040 C27SQX 46879964 EC50 = 3700 nM T84040 CVTM60 46879965 EC50 = 1000 nM T84040 C2TCG9 46880022 EC50 > 25000 nM T84040 CPH2B0 46880023 EC50 > 25000 nM T84040 C0DPM5 46880024 EC50 > 25000 nM T84040 CM79PR 46880025 EC50 > 25000 nM T84040 CQ8CZ3 46880026 EC50 > 25000 nM T84040 C2PQ6Z 46880080 EC50 > 25000 nM T84040 CA0S7Z 46880081 EC50 > 25000 nM T84040 C3F9BQ 46880082 EC50 > 25000 nM T84040 CA90CL 46889923 EC50 = 0.5754 nM T84040 C3TK9C 46889974 EC50 = 200 nM T84040 CJR0H1 46889975 EC50 = 130 nM T84040 CWB6N9 46889990 EC50 = 1200 nM T84040 CMEW07 46889991 IC50 < 1000 nM T84040 CUC71M 46889992 IC50 < 1000 nM T84040 C19QAB 46890000 EC50 = 660 nM T84040 C29WDK 46890001 EC50 = 3760 nM T84040 CJRY52 46890002 EC50 = 4630 nM T84040 CR25IP 46890003 EC50 = 5650 nM T84040 C0ULH8 46890004 EC50 = 0.4 nM T84040 CS9D5Y 46890005 IC50 = 1100 nM T84040 C70HJR 46947247 IC50 = 1300 nM T84040 C46KOW 49780146 EC50 = 1.6 nM T84040 C5LKC0 49780147 EC50 = 0.1 nM T84040 C7I3OT 49780151 EC50 = 7.7 nM T84040 CCK52O 49783411 EC50 = 33 nM T84040 CWD2X1 49783412 EC50 = 3.5 nM T84040 CDP79Z 49783413 EC50 = 158 nM T84040 CR63FA 51039271 IC50 = 10 nM T84040 C5DBY8 53348079 IC50 > 32000 nM T84040 C3OBC9 56666148 EC50 = 49 nM T84040 C0EY9W 56673065 EC50 = 27 nM T84040 C60YJB 56673066 EC50 = 109 nM T84040 CA0DR5 56683038 EC50 = 79 nM T84040 CA65JN 56951566 IC50 = 85 nM T84040 CR9Z7B 57345605 IC50 = 400 nM T84040 CUZ9F0 57392692 IC50 = 4100 nM T84040 CUWP23 57393398 IC50 = 3700 nM T84040 C1WJ7G 57395139 IC50 = 1800 nM T84040 C6MP0B 57396031 IC50 = 2600 nM T84040 CP1SY0 57396893 IC50 = 1100 nM T84040 C23TSZ 57396906 IC50 = 3100 nM T84040 C9L8OW 57400322 IC50 = 3100 nM T84040 CD9MH8 57403002 IC50 = 2100 nM T84040 C4KHD7 57403874 IC50 = 1600 nM T84040 CK5XR1 60020772 IC50 > 32000 nM T84040 C42XKO 60023185 IC50 > 32000 nM T84040 CO8PX6 60023237 IC50 = 3200 nM T84040 CC58DQ 60023252 IC50 > 32000 nM T84040 CPO5E1 60023291 IC50 > 32000 nM T84040 CYU13V 66832911 IC50 = 154 nM T84040 CYZ29G 68817251 EC50 > 30000 nM T84040 CX5W2A 70682601 IC50 = 251.19 nM T84040 C7Q4EF 70682602 IC50 = 5011.87 nM T84040 CTBU29 70682603 IC50 = 398.11 nM T84040 CV1F8K 70682604 IC50 = 3981.07 nM T84040 CP01WE 70682605 IC50 = 1584.89 nM T84040 CD9ZK1 70682606 IC50 = 1000 nM T84040 CUS4K8 70684696 IC50 = 398.11 nM T84040 C01RLE 70684697 IC50 = 794.33 nM T84040 C6Q1KL 70684698 IC50 = 199.53 nM T84040 C6K1RJ 70684699 IC50 = 398.11 nM T84040 CV1R8A 70688913 IC50 = 3981.07 nM T84040 COVK93 70688915 IC50 = 3162.28 nM T84040 CJLX93 70688916 IC50 = 1584.89 nM T84040 CC58EF 70688920 IC50 = 5011.87 nM T84040 CY78WT 70688921 IC50 = 3981.07 nM T84040 C9LQ4T 70688922 IC50 = 10 nM T84040 CM18JP 70691008 IC50 = 1000 nM T84040 CG4RD0 70693133 IC50 = 398.11 nM T84040 C0ZGV3 70693134 IC50 = 3981.07 nM T84040 C6J1XH 70693138 IC50 = 251.19 nM T84040 CP5VG7 70693139 IC50 = 1258.93 nM T84040 CQ06EC 70695195 IC50 = 1258.93 nM T84040 CMXL57 70695196 IC50 = 6309.57 nM T84040 CH3LO9 70695197 IC50 = 2511.89 nM T84040 C3M5FQ 70695198 IC50 = 3162.28 nM T84040 C67ZOE 70695199 IC50 = 1995.26 nM T84040 CFD97I 70695205 IC50 = 6309.57 nM T84040 C82EHB 70695206 IC50 = 1995.26 nM T84040 CR47JE 70695208 IC50 = 3162.28 nM T84040 CG7D3B 70697238 IC50 = 501.19 nM T84040 CDU5F2 70697242 IC50 = 2511.89 nM T84040 CY2ON5 70697243 IC50 = 5011.87 nM T84040 CU4Z3G 71582398 EC50 = 19100 nM T84040 CW20HQ 71818431 IC50 = 8000 nM T84040 C2L7TX 71818575 IC50 = 25000 nM T84040 CA9CX5 72197094 EC50 = 150 nM T84040 CV6ZT3 73297271 IC50 = 131 nM T84040 CEZK64 90645309 IC50 = 310 nM T84040 CXUH46 90645310 IC50 = 320 nM T84040 C0NM1C 90645311 IC50 = 330 nM T84040 CL0O7Q 90645312 IC50 = 410 nM T84040 C75ORJ 90645313 IC50 = 630 nM T84040 C8J7DS 90645314 IC50 = 630 nM T84040 CYOH25 90645315 IC50 = 650 nM T84040 C1KS5J 90645316 IC50 = 710 nM T84040 C8S1XM 90645317 IC50 = 1100 nM T84040 C9FC7Q 90645318 IC50 = 1100 nM T84040 C3J5KC 90645319 IC50 = 1200 nM T84040 CE91HF 90645320 IC50 = 1200 nM T84040 C1JTK3 90645321 IC50 = 1300 nM T84040 CVM1A8 90645322 IC50 = 1600 nM T84040 CO6ZX3 90645323 IC50 = 2000 nM T84040 CH2BF1 90645324 IC50 = 2200 nM T84040 CBXM40 90645325 IC50 = 2500 nM T84040 C7TL0Y 90645326 IC50 = 2700 nM T84040 CJEZ93 90645327 IC50 = 3000 nM T84040 C0Z1LE 90645328 IC50 = 3000 nM T84040 C5FWV7 90645329 IC50 = 3100 nM T84040 C9LWH6 90645330 IC50 > 32000 nM T84040 C2A3ED 90645331 IC50 > 32000 nM T84040 C9Q3ME 90645332 IC50 > 32000 nM T84040 C87KCZ 90645333 IC50 > 32000 nM T84040 C7TPE8 90645334 IC50 > 32000 nM T84040 CEJ40C 90645335 IC50 > 32000 nM T84040 CUFM82 90645336 IC50 > 32000 nM T84040 CL3X5T 90645337 IC50 > 32000 nM T84040 CDVG72 90645338 IC50 > 32000 nM T84040 CG41MW 90645339 IC50 > 32000 nM T84040 CBM4W1 90645340 IC50 > 32000 nM T84040 C61XTZ 90645341 IC50 > 32000 nM T84040 C8HDR4 90645342 IC50 > 32000 nM T84040 C7X9ZK 90645343 IC50 > 32000 nM T84040 CW7AZ5 90645441 IC50 = 1230 nM T84040 CC0M7F 90645442 IC50 = 3950 nM T84040 CRB14Q 90645443 IC50 = 7810 nM T84040 C3UH2Q 90645444 IC50 = 584 nM T84040 CSG79U 90645445 IC50 = 514 nM T84040 CJ1VR3 90645446 IC50 = 3400 nM T84040 CN61RW 90645447 IC50 = 84 nM T84040 CAF23J 90645448 IC50 = 2200 nM T84040 C4N3VR 90645449 IC50 = 3430 nM T84040 CVJ8F1 90645450 IC50 = 8900 nM T84040 C06JXN 90645451 IC50 = 30000 nM T84040 C41IRH 90645452 IC50 = 306 nM T84040 CMTN81 90645453 IC50 = 1230 nM T84040 CRZ6X3 90645454 IC50 = 296 nM T84040 CTP6C7 90645455 IC50 = 48 nM T84040 C90KGC 90645456 IC50 = 3090 nM T84040 CERN74 90645457 IC50 = 6720 nM T84040 C9DX0Y 90645458 IC50 = 7410 nM T84040 CISP03 90645459 IC50 = 24 nM T84040 CM5FN9 90645460 IC50 = 15 nM T84040 CL5TV9 90645461 IC50 = 50 nM T84040 C7Q5FW 90645462 IC50 = 25400 nM T84040 CNQS85 90645463 IC50 = 61 nM T84040 CI6TW7 90645464 IC50 = 103 nM T84040 C31TXQ 90645465 IC50 = 26 nM T84040 CDK3T1 90645466 IC50 = 39 nM T84040 CYR82I 90645467 IC50 = 970 nM T84040 C6OF3B 90645468 IC50 = 26 nM T84040 C9J5TE 90645469 IC50 = 142 nM T84040 C0VW1K 90645470 IC50 = 36 nM T84040 CAG1Q0 90645471 IC50 = 50 nM T84040 C3BV7M 90645472 IC50 = 129 nM T84040 CXC74T 90645473 IC50 > 30000 nM T84040 C6SU4X 90665452 IC50 > 12500 nM T84040 CJCR26 90665456 EC50 > 12500 nM T84040 C40TVU 90667106 IC50 = 100 nM T84040 C1WTS6 90667107 IC50 = 150 nM T84040 CRN34L 90667108 IC50 = 200 nM T84040 C7P3NV 90667109 IC50 = 200 nM T84040 C5GJ2Z 90667110 IC50 = 400 nM T84040 C57QGM 118008139 IC50 = 1200 nM T84040 CKV54B 118008525 IC50 = 4400 nM T84040 C08HJA 118019699 IC50 = 69 nM T84040 CPG3D6 118019741 IC50 = 239 nM T84040 CPT09N 118019761 IC50 = 1500 nM T84040 C10YVO 118019777 IC50 = 13 nM T84040 CDNC39 118246723 EC50 > 30000 nM T84040 C4A7GI 118707060 IC50 = 2700 nM T84040 C1IKV3 118707061 IC50 = 2900 nM T84040 C0PQ8W 118707062 IC50 = 3900 nM T84040 CEO1U0 118707063 IC50 = 2300 nM T84040 C7GBV6 118707064 IC50 > 32000 nM T84040 CD4JK0 118707065 IC50 = 1300 nM T84040 C8T7MK 118707066 IC50 = 790 nM T84040 CONA71 118707067 IC50 = 390 nM T84040 C9J1MO 118707068 IC50 = 290 nM T84040 CQI54L 118707069 IC50 = 200 nM T84040 C2WLS7 118707070 IC50 > 32000 nM T84040 CCWU94 118707071 IC50 = 940 nM T84040 C2FSQ8 118707072 IC50 = 2600 nM T84040 C0C4TQ 118707073 IC50 = 1400 nM T84040 C2U3CZ 118707074 IC50 = 1200 nM T84040 CTXH13 118707075 IC50 = 110 nM T84040 CH0BJ1 118707076 IC50 > 32000 nM T84040 CN2I1Q 118707077 IC50 = 74 nM T84040 CK1FR6 118707078 IC50 = 91 nM T84040 C6EJT4 118707079 IC50 > 32000 nM T84040 COQ2G7 118707080 IC50 > 32000 nM T84040 CLJ9E5 118707081 IC50 = 1900 nM T84040 CEC73B 118707619 IC50 > 2000 nM T84040 CGF16J 118707620 IC50 = 1200 nM T84040 C6U5YJ 118707621 EC50 > 40000 nM T84040 C8AP1E 118707622 IC50 = 970 nM T84040 CXE02U 118707623 IC50 = 710 nM T84040 CVW24U 118707624 IC50 = 300 nM T84040 C6PI3N 118707625 IC50 = 590 nM T84040 CI32HS 118707626 IC50 = 200 nM T84040 CU06CA 118707627 IC50 = 170 nM T84040 CXH60W 118707628 IC50 = 940 nM T84040 C9MB7E 118707629 IC50 > 40000000 nM T84040 CZH02O 118711168 EC50 = 26000 nM T84040 C0QMH8 121304823 IC50 = 1 nM T84040 C9F2WA 121304824 IC50 = 1900 nM T84040 C6C9EF 121304827 IC50 = 0.7 nM T84040 C74PDS 121304861 IC50 = 73 nM T84040 CI7C4R 121304866 IC50 = 63 nM T84040 CK2U7O 121313637 IC50 = 12 nM T84040 C3H7EJ 121313649 IC50 = 309 nM T84040 C4FL6N 121313654 IC50 = 91 nM T84040 CD2C0X 122489185 IC50 = 5 nM T84040 CV95GP 122489372 IC50 = 179 nM T84040 C6R2KP 122489391 IC50 = 64 nM T84040 C4IA5J 122489392 IC50 = 5 nM T84040 CA5HR7 122489394 IC50 = 8 nM T84040 CDA78U 122489431 IC50 = 10 nM T84040 COJ90L 122490037 IC50 = 96 nM T84040 CN0R4Z 122490110 IC50 = 184 nM T84040 C1R4IV 122490118 IC50 = 13 nM T84040 CMP5Z4 122534006 IC50 = 33 nM T84040 C1O6RC 122534008 IC50 = 113 nM T84040 CU4O0B 126752051 IC50 = 153 nM T84040 C0K2CR 127030063 IC50 = 1180 nM T84040 CCK2N4 127030939 IC50 = 918 nM T84040 CWE8M1 127031838 IC50 = 41 nM T84040 CN0C1X 127031917 IC50 = 165 nM T84040 C0ZKU5 127031918 IC50 = 63 nM T84040 C3W5YJ 127032100 IC50 = 136 nM T84040 CX9M5R 127032469 IC50 = 286 nM T84040 CN5WY4 127032470 IC50 = 1330 nM T84040 C1CDB0 127032471 IC50 = 1460 nM T84040 C5JYL1 127032762 IC50 = 265 nM T84040 CE3ZQ9 127032763 IC50 = 70 nM T84040 CD7N2R 127032770 IC50 = 201 nM T84040 CKPD15 127032771 IC50 = 1710 nM T84040 CA76JT 127032772 IC50 = 1580 nM T84040 C2UC8N 127032773 IC50 = 41 nM T84040 CPD5K3 127032784 IC50 > 16700 nM T84040 CGXS84 127032785 IC50 > 4200 nM T84040 CK7M9I 127033094 IC50 = 2180 nM T84040 C1BXG8 127033365 IC50 = 16 nM T84040 CK1X5L 127033366 IC50 = 211 nM T84040 C2BVC1 127034205 IC50 = 52 nM T84040 C9G0VT 127034206 IC50 = 2120 nM T84040 CUBE39 127034207 IC50 = 58 nM T84040 C9W5AH 127034465 IC50 = 150 nM T84040 C9CY5F 127034466 IC50 = 933 nM T84040 CKV35Q 127034467 IC50 = 85 nM T84040 C4SKV2 127036380 IC50 = 20 nM T84040 CZ7DU5 127036381 IC50 = 380 nM T84040 CL25MU 127036570 IC50 = 130 nM T84040 CLE41K 127036571 IC50 = 110 nM T84040 CGQ18L 127036793 IC50 > 20000 nM T84040 CL70HX 127037222 IC50 = 23 nM T84040 C0W7VU 127037223 IC50 = 63 nM T84040 CH4BK9 127037224 IC50 = 270 nM T84040 C2WR8Z 127037225 IC50 > 20000 nM T84040 CH1J2T 127037226 IC50 > 18000 nM T84040 CL7YG9 127037246 IC50 > 20000 nM T84040 COF6E5 127037247 IC50 > 20000 nM T84040 CKS0A3 127037248 IC50 > 20000 nM T84040 CY71EX 127037249 IC50 = 6700 nM T84040 C3XV1S 127037389 IC50 > 19000 nM T84040 CW87KJ 127037390 IC50 = 290 nM T84040 C08BEP 127037391 IC50 = 190 nM T84040 CCNO28 127037449 IC50 = 350 nM T84040 CP19BC 134134923 IC50 = 2 nM T84040 CS5ZL7 134141534 IC50 = 43 nM T84040 CTM36F 134154327 IC50 = 7 nM T84040 C8LQY2 134157451 IC50 = 4 nM T84040 C3TW0A 134374895 IC50 > 30000 nM T84040 CCJ09K 136002659 EC50 = 2.1 nM T84040 C73FQR 137631928 IC50 = 257 nM T84040 CHQN12 137632885 IC50 = 2537 nM T84040 CG5IH6 137633289 IC50 > 10000 nM T84040 C8USM4 137635104 IC50 = 74 nM T84040 C5N0HL 137635177 IC50 = 131 nM T84040 C7VN4C 137636068 IC50 = 328 nM T84040 COE98I 137636816 IC50 = 1203 nM T84040 C8Y2CR 137637063 IC50 = 2100 nM T84040 CJH2V9 137637559 IC50 = 20 nM T84040 C63PMN 137639029 IC50 > 10000 nM T84040 CZE78F 137640208 IC50 = 645 nM T84040 CX81RJ 137641194 IC50 = 134 nM T84040 CTZ0G6 137642738 IC50 = 111 nM T84040 C2N7VF 137642995 IC50 = 2300 nM T84040 CACN52 137643000 EC50 > 30000 nM T84040 C8ER3H 137646167 IC50 = 11700 nM T84040 CW0O9Z 137646494 IC50 = 3700 nM T84040 COH13Y 137647733 IC50 = 1182 nM T84040 C3JH7F 137651968 IC50 > 10000 nM T84040 CD2U6O 137652413 IC50 = 4630 nM T84040 CJA30D 137652497 IC50 = 2667 nM T84040 CL8K6R 137652927 IC50 = 42 nM T84040 CV1W8A 137653423 IC50 = 91 nM T84040 CF42SD 137653875 IC50 > 20000 nM T84040 CU4N6L 137656453 IC50 = 38 nM T84040 CXAQ20 137657618 IC50 > 10000 nM T84040 CJET49 137658836 IC50 = 748 nM T84040 CJ9N2I 137659640 IC50 = 450 nM T84040 CJE64C 137659970 IC50 = 53 nM T84040 C2KX3V 137661020 IC50 = 686 nM T84040 CEK6B1 139300630 IC50 > 10000 nM T84040 C25MLZ 145963901 IC50 > 10000 nM T84040 C10KZD 145963912 IC50 > 1000 nM T84040 CR0SM9 145964107 IC50 = 71 nM T84040 C97SAY 145964896 IC50 = 474 nM T84040 CVX41T 145965582 IC50 = 53 nM T84040 C2EY5H 145965868 IC50 > 10000 nM T84040 CM2X3D 145966564 IC50 = 159 nM T84040 CM72AJ 145970513 IC50 = 1451 nM T84040 C3JB7Y 145971661 IC50 > 10000 nM T84040 CK7M8X 145972092 IC50 = 1900 nM T84040 CKV69S 145972153 IC50 > 1000 nM T84040 CI9UB1 145973068 IC50 = 673 nM T84040 CJ7ID8 145974237 IC50 > 3000 nM T84040 C74VRF 145974399 IC50 > 10000 nM T84040 CQM72A 145974444 IC50 = 1000 nM T84040 CS06GB 145974517 IC50 > 3000 nM T84040 COM5P8 145974902 IC50 = 1700 nM T84040 CO2XP9 145974914 IC50 > 10000 nM T84040 CU36PQ 145975340 IC50 > 10000 nM T84040 C89OFN 145975833 IC50 > 10000 nM T84040 C8L7JG 145976550 IC50 = 101 nM T84040 C5L1NO 145976862 IC50 > 1000 nM T84040 CYNU62 145977293 IC50 = 851 nM T84040 CH6N2Z 145977445 IC50 = 83 nM T84040 C65GEI 145977562 IC50 = 825 nM T84040 C7YJG8 145978486 IC50 = 26700 nM T84040 C7YM1K 155527804 EC50 = 11000 nM T84040 CVC46M 155555048 IC50 = 100000 nM T84040 CE2G6O 135870665 IC50 = 8610 nM T84040 CC8T4B 26487 EC50 = 15100 nM T84040 C8KF3N 35020890 EC50 = 22400 nM T84040 D00AJB 73255 EC50 = 8000 nM T84040 D00AVT 16441 EC50 = 41000 nM T84040 D00TWK 185914 EC50 > 30000 nM T84040 D01PGU 5311211 EC50 = 5600 nM T84040 D01RPM 11645581 EC50 = 1000 nM T84040 D01RUO 10878016 EC50 = 3 nM T84040 D03GXQ 3727 EC50 = 357000 nM T84040 D03LVI 2830271 IC50 = 35 nM T84040 D03LVL 53464483 IC50 > 25000 nM T84040 D04NOT 11715 EC50 = 1100 nM T84040 D04ULU 161930 EC50 = 100000 nM T84040 D04XXE 73489 EC50 = 16000 nM T84040 D05CRM 3277297 IC50 = 120 nM T84040 D05DTN 6445537 EC50 = 1900 nM T84040 D06OLJ 3089985 IC50 = 28 nM T84040 D07JDC 10364 EC50 = 7000 nM T84040 D07LNY 5280880 EC50 = 24000 nM T84040 D08DQL 4549 EC50 = 320 nM T84040 D08MUZ 5364752 EC50 = 5000 nM T84040 D09CSB 447466 EC50 = 16000 nM T84040 D0A1UL 49783953 IC50 > 10000 nM T84040 D0D6MC 1150897 IC50 = 1800 nM T84040 D0G4GB 10757 EC50 = 30 nM T84040 D0I0AA 7847 EC50 = 800 nM T84040 D0J0BV 2873523 IC50 = 14300 nM T84040 D0K6RG 7498 EC50 = 12000 nM T84040 D0MZ7C 37839 EC50 = 590 nM T84040 D0N3CZ 12480411 EC50 = 800 nM T84040 D0N7MS 5353376 EC50 = 28000 nM T84040 D0NH1E 1383884 EC50 = 100 nM T84040 D0O3FC 2830270 IC50 = 29 nM T84040 D0P0IE 10205 EC50 = 460 nM T84040 D0P7VQ 9929425 EC50 = 4500 nM T84040 D0PJ3M 637511 EC50 = 6500 nM T84040 D0S2GF 17604 EC50 = 0.9 nM T84040 D0V8DH 53380803 EC50 = 23 nM T84040 D0X9YD 65036 EC50 = 1910 nM T21669 D02TQO 14985 IC50 = 500 nM T21669 D06TNL 3278 IC50 = 3400 nM T21669 CZA12R 5141 Ki = 10000 nM T21669 CM1IT6 27815 IC50 = 600 nM T21669 CL3OU2 122297 IC50 = 51.2 nM T21669 CDP49B 157619 Ki = 490 nM T21669 C6GBA8 313611 IC50 = 1000 nM T21669 CG4P6H 4411483 IC50 > 250000 nM T21669 C0ZFP5 6439061 IC50 = 13200 nM T21669 C2J0YM 9817686 IC50 = 800 nM T21669 C3IR7T 10422367 Ki = 123900 nM T21669 C5QFS8 10447087 Ki = 6100 nM T21669 C6JY9S 11346229 IC50 = 1400 nM T21669 C1N8QB 11743150 Ki = 40000 nM T21669 C34KBV 13745578 IC50 = 3100 nM T21669 CKY6D4 13885287 Ki = 1110 nM T21669 CXP1S2 14132141 Ki = 187000 nM T21669 CJ8E1F 17980079 IC50 >= 100000 nM T21669 CHX0E8 20731911 Ki = 420 nM T21669 CYDF65 25019607 IC50 = 5000 nM T21669 C4D1IP 25019608 IC50 = 1970 nM T21669 CKT7I0 25019609 IC50 = 4000 nM T21669 C4GAJ8 25019869 IC50 = 1800 nM T21669 C3ON1V 25019870 IC50 = 2100 nM T21669 CP47XA 25019871 IC50 = 600 nM T21669 CA4IN2 25019874 IC50 = 3200 nM T21669 CCA7U6 25019875 IC50 = 2000 nM T21669 CF17BR 44300879 Ki = 550000 nM T21669 CEWB31 44300893 Ki = 850 nM T21669 COJ56C 44300905 Ki = 120 nM T21669 C3TXO9 44300921 Ki = 710000 nM T21669 C06ENG 44385619 IC50 = 217000 nM T21669 CAZ2K0 44385682 IC50 > 250000 nM T21669 C7HWG6 44385932 IC50 = 5200 nM T21669 CQ7V5J 44386040 IC50 > 250000 nM T21669 C6IM9P 44386041 IC50 = 155000 nM T21669 CAGC58 44386723 IC50 = 8100 nM T21669 C0W2HB 44386941 IC50 = 40300 nM T21669 CIS37G 44386993 IC50 > 250000 nM T21669 CS9HI5 44387048 IC50 = 208000 nM T21669 C3G1TO 44387218 IC50 > 250000 nM T21669 C7U4IO 44403943 Ki = 660 nM T21669 CH8DC4 44404193 IC50 = 10800 nM T21669 C2PJ1R 44413511 IC50 = 15046 nM T21669 COH04A 44413512 IC50 = 992.4 nM T21669 C5UL0A 44413513 IC50 = 704 nM T21669 CIB79M 44413514 IC50 = 1022 nM T21669 CYR90A 44413516 IC50 = 624 nM T21669 C1YL6S 44413517 IC50 = 46.1 nM T21669 CY14GT 44413518 IC50 = 31 nM T21669 C7L1EF 44413967 IC50 = 142 nM T21669 CY0KD5 44597665 IC50 > 100000 nM T21669 CESJ03 45484201 IC50 = 2300 nM T21669 CTLQ36 45484202 IC50 = 1300 nM T21669 C1LTE4 45484207 IC50 = 3500 nM T21669 C06MSW 45484217 IC50 = 700 nM T21669 C69XVG 45484220 IC50 = 3300 nM T21669 CU19ZF 45484221 IC50 = 2400 nM T21669 CAWL21 45484226 IC50 = 700 nM T21669 C7NLX1 45484227 IC50 = 4000 nM T21669 CVO19L 45484234 IC50 = 3600 nM T21669 C9ABC5 45484241 IC50 = 2900 nM T21669 C2QUS4 45484242 IC50 = 3900 nM T21669 CEY7K9 45484248 IC50 > 40000 nM T21669 CP1A3N 45484253 IC50 = 3800 nM T21669 CYE24A 45484257 IC50 = 3900 nM T21669 CZQB96 45484258 IC50 = 5400 nM T21669 CEQR23 45484259 IC50 = 3300 nM T21669 CT3IL8 45484276 IC50 = 2000 nM T21669 COAS69 45484285 IC50 = 1400 nM T21669 CP1YM8 56926704 IC50 > 100000 nM T21669 CKR36B 56926707 IC50 > 100000 nM T21669 C0IV7W 56926708 IC50 > 100000 nM T21669 CVH3P7 56926709 IC50 = 24500 nM T21669 CV67LZ 56926804 IC50 = 82500 nM T21669 CK93PW 56926805 IC50 = 62700 nM T21669 CYC1M7 56926806 IC50 = 20200 nM T21669 CQH63T 56926807 IC50 = 48200 nM T21669 C2VQ0R 56926808 IC50 = 37600 nM T21669 C98YWR 56926809 IC50 = 52400 nM T21669 C40ALR 56926915 IC50 = 179000 nM T21669 C40KLT 56926916 IC50 = 58000 nM T21669 CQXL53 56926917 IC50 = 186700 nM T21669 C0C9PN 56926918 IC50 = 36500 nM T21669 CFK43A 79682737 IC50 = 7400 nM T21669 CD3KV5 85813946 IC50 = 1700 nM T21669 CLP62N 118724259 IC50 = 200 nM T21669 C18FIR 118724260 IC50 = 500 nM T21669 CT72ZS 118724261 IC50 = 1400 nM T21669 CNWA46 118724262 IC50 = 1800 nM T21669 CTI89N 118724263 IC50 = 800 nM T21669 CF62OM 118724265 IC50 = 600 nM T21669 CLY76V 118724266 IC50 = 500 nM T21669 C21AZU 118724267 IC50 = 1200 nM T21669 C3PJ6M 118724268 IC50 = 1000 nM T21669 CAT5C4 118724269 IC50 = 2100 nM T21669 CA56BS 118724270 IC50 = 1000 nM T21669 CA1D9C 118724271 IC50 = 400 nM T21669 C3FH4N 118724272 IC50 = 700 nM T21669 CB86LE 118724273 IC50 = 100 nM T21669 C6W7ZP 118724274 IC50 = 1600 nM T21669 CNE3F5 118724275 IC50 = 700 nM T21669 CAM0S3 118724276 IC50 = 200 nM T21669 C5AP6T 118724277 IC50 = 100 nM T21669 CG63AT 118724278 IC50 = 1700 nM T21669 CKW14F 118724279 IC50 = 1800 nM T21669 CR90AJ 118724280 IC50 = 6900 nM T21669 C5RZ7H 118724281 IC50 = 4800 nM T21669 C18WEV 118724282 IC50 = 6500 nM T21669 C1Q0LU 118724283 IC50 = 600 nM T21669 C82VQF 118724284 IC50 = 400 nM T21669 CW0PU6 118724285 IC50 = 300 nM T21669 C30RBO 118724286 IC50 = 300 nM T21669 C52ZDU 118724287 IC50 = 500 nM T21669 C8EDZ1 118724288 IC50 = 14000 nM T21669 CL1ZR5 118724289 IC50 = 9000 nM T21669 CYZ6Q3 118724290 IC50 >= 100000 nM T21669 C3B4VU 135426515 IC50 = 35700 nM T21669 C2APM1 135453064 IC50 = 35100 nM T21669 CXW57D 135862918 IC50 = 2100 nM T21669 C75KBI 135862919 IC50 = 3400 nM T21669 CP2Q6W 136087118 IC50 = 1200 nM T21669 D0A1CM 5281855 IC50 = 77100 nM T34843 CX7S0D 70683012 EC50 = 0.09 nM T34843 CTH8D2 127048230 EC50 = 8.1 nM T34843 C6IME2 127048235 EC50 = 0.09 nM T34843 CYQ06U 127048242 EC50 = 0.2 nM T34843 CSJ4E0 127048563 EC50 = 0.14 nM T34843 C06PAY 127048570 EC50 = 0.66 nM T34843 CIC5N9 127048573 EC50 = 0.06 nM T34843 C0QD6C 127048580 EC50 = 0.11 nM T34843 COAX23 127048585 EC50 = 0.13 nM T34843 C9AYL1 127048586 EC50 = 0.05 nM T34843 CQJ4I9 127048907 EC50 = 0.11 nM T34843 CNFT67 127048913 EC50 = 0.15 nM T34843 C2T1RK 127048919 EC50 > 30 nM T34843 CZM2P6 127048924 EC50 = 0.11 nM T34843 CU6B7T 127048925 EC50 = 0.51 nM T34843 C9CBY0 127049246 EC50 = 0.08 nM T34843 C3EZ1Q 127049553 EC50 = 0.23 nM T34843 CHF48Z 127049554 EC50 = 7.1 nM T34843 CZ04YP 127049559 EC50 = 0.35 nM T34843 CF8E4Y 127049561 EC50 = 0.11 nM T34843 CTND43 127049562 EC50 = 0.03 nM T34843 C2YK9U 127049569 EC50 = 0.1 nM T34843 CU0WT7 127049891 EC50 = 0.07 nM T34843 C8O3ZH 127049892 EC50 = 2.6 nM T34843 C91XKU 127049900 EC50 = 1.1 nM T34843 C91XMF 127049904 EC50 = 1.5 nM T34843 C05KIM 127049905 EC50 = 0.47 nM T34843 CGZI28 127049907 EC50 = 0.09 nM T34843 CI3X9N 127050190 EC50 = 0.1 nM T34843 CJ8MO0 127050192 EC50 = 0.29 nM T34843 CLQE96 127050193 EC50 = 2.2 nM T34843 C2T3NQ 127050489 EC50 = 0.22 nM T34843 C52ROH 127050497 EC50 = 0.44 nM T34843 CUY7X9 127050499 EC50 = 0.31 nM T34843 C6X9AW 127050816 EC50 = 0.03 nM T34843 CJ79TN 127050817 EC50 = 4.5 nM T34843 CQKE41 127050829 EC50 = 0.03 nM T34843 C6VX5B 127051083 EC50 = 0.05 nM T34843 CO0MQ4 127051084 EC50 = 1.9 nM T34843 CCVE81 127051086 EC50 = 0.15 nM T34843 C1URK5 127051088 EC50 = 1.5 nM T34843 CG4D0F 127051089 EC50 = 0.06 nM T34843 CQT03Z 127051091 EC50 = 0.07 nM T34843 C8AWI0 127051094 EC50 = 4.5 nM T34843 COS48H 127051377 EC50 = 0.48 nM T34843 CX8AU4 127051382 EC50 = 16 nM T34843 C21PCY 127051386 EC50 = 0.2 nM T34843 CYN56P 127051391 EC50 > 30 nM T34843 C97SOU 127051393 EC50 = 0.06 nM T34843 CG7W2D 127051708 EC50 = 0.1 nM T34843 CV96NH 127051710 EC50 = 0.1 nM T34843 CQ7G8U 127051715 EC50 = 0.09 nM T34843 CAJ0F5 127051716 EC50 = 0.15 nM T34843 CZL51Q 127051717 EC50 = 0.04 nM T34843 C2AWU3 127051718 EC50 = 0.08 nM T34843 CK41ZJ 127052018 EC50 = 8.9 nM T34843 CS0HY2 127052019 EC50 = 0.21 nM T34843 CE63MT 127052022 EC50 = 1.1 nM T34843 CC7DM5 127052029 EC50 = 0.18 nM T34843 C4PO0G 127052034 EC50 = 0.42 nM T34843 C5CUZ1 127052341 EC50 = 0.16 nM T34843 C9QC7T 127052344 EC50 = 0.2 nM T34843 C95WZR 127052351 EC50 = 0.07 nM T34843 CKQG87 127052643 EC50 = 0.19 nM T34843 CAO0W7 127052645 EC50 = 0.03 nM T34843 CN0LF8 127052647 EC50 = 0.43 nM T34843 C0I1LV 127052648 EC50 = 0.63 nM T34843 CW4V7K 127052654 EC50 = 0.04 nM T34843 C5K3JR 127052936 EC50 = 0.08 nM T34843 CXJ7C0 127052938 EC50 = 14 nM T34843 C3RTO1 127052943 EC50 = 0.09 nM T34843 C75QMW 127052944 EC50 = 0.13 nM T34843 CY9L1H 127052945 EC50 = 0.38 nM T34843 COB7C9 127052953 EC50 = 0.09 nM T34843 CU1P4W 145948755 EC50 = 0.51 nM T34843 CGY3Q0 145948765 EC50 = 0.22 nM T34843 CAXE41 145948867 EC50 = 0.1 nM T34843 CB3D9P 145948868 EC50 = 0.13 nM T34843 CR2M7E 145948881 EC50 = 0.18 nM T34843 CIDG54 145948888 EC50 = 0.13 nM T34843 CZ70FB 145948890 EC50 = 0.16 nM T34843 CTV1K7 145948929 EC50 = 0.29 nM T34843 CQ6I0F 145948972 EC50 = 0.19 nM T34843 C5QB1Z 145948975 EC50 = 0.35 nM T34843 C1XVJ3 155547905 EC50 = 0.09 nM T34843 CS8BW0 155560523 EC50 = 1 nM T49755 C67ACJ 127025037 IC50 = 3770 nM T49755 CJ1I3R 127025355 IC50 = 4710 nM T49755 C7QS3P 127025356 IC50 = 4870 nM T49755 C2SH1G 127025357 IC50 = 4330 nM T49755 C9N3HW 127025635 IC50 = 5500 nM T49755 CLR2T9 127025636 IC50 = 4060 nM T49755 CN0WF5 127025924 IC50 = 3740 nM T49755 CE3T1M 127025925 IC50 = 4610 nM T49755 CMRG93 127026221 IC50 = 3380 nM T49755 CAD78W 127027122 IC50 = 5230 nM T49755 CDA2K7 127027123 IC50 = 6160 nM T49755 C65XFO 127040605 IC50 = 3000 nM T56496 CLZA82 1215 Ki = 90 nM T56496 CS46QU 7408 Ki = 830000 nM T56496 C6RVS2 17535 Ki = 14800 nM T56496 C51OJF 27697 Ki = 51000 nM T56496 CR0I2T 34005 Ki = 450000 nM T56496 CT80UY 66648 IC50 = 20000 nM T56496 CC3FE1 75818 Ki = 430000 nM T56496 C4FXT6 77802 IC50 = 9000 nM T56496 C7V4FT 93889 Ki = 730000 nM T56496 C98SWZ 116521 Ki = 300000 nM T56496 CYHJ29 123919 Ki = 3 nM T56496 CCQ34V 217958 IC50 = 20000 nM T56496 CI6J5L 587625 IC50 = 600 nM T56496 CAY2G6 643189 Ki = 4800000 nM T56496 CLV0B1 2776381 Ki = 110000 nM T56496 CBM52Z 3085076 Ki = 37000 nM T56496 C6AML5 5288606 Ki = 40 nM T56496 CA3XE0 10019263 Ki = 130 nM T56496 C0J3PI 10089519 Ki = 1 nM T56496 CFZN32 10108068 Ki = 1700 nM T56496 CZ3RL4 10176243 Ki = 1500 nM T56496 C0Z3NS 10263132 Ki = 10000 nM T56496 C9FDM0 10263774 Ki = 52 nM T56496 CVJ78Z 10331921 Ki = 2000 nM T56496 C3NGO6 10332138 Ki = 2300 nM T56496 CB6HO1 10377457 Ki = 67 nM T56496 CM7D5X 10399576 Ki = 150 nM T56496 C8OZ2X 10401405 Ki = 3200 nM T56496 CPR21Q 10425899 Ki = 560 nM T56496 CRX56L 10471609 Ki = 61 nM T56496 CR20KW 10487987 Ki = 1600 nM T56496 C1PFR6 10514405 Ki = 1200 nM T56496 COCQ40 10562109 Ki = 1100 nM T56496 C1JH8P 10565477 Ki = 70 nM T56496 C5SX1B 10588353 Ki = 9000 nM T56496 CV94SO 10607760 Ki = 16 nM T56496 C5VS4G 10610245 Ki = 1100 nM T56496 CQML32 10618144 Ki = 610 nM T56496 CT9Q0C 10632080 Ki = 3500 nM T56496 CT30XH 10634951 Ki = 3700 nM T56496 C32HNJ 10711778 Ki = 26000 nM T56496 C4VK0T 10729255 Ki = 56 nM T56496 C04RAP 10733711 Ki = 23000 nM T56496 C8WEF4 10736630 Ki = 6300 nM T56496 CY1S0D 10750185 Ki = 2600 nM T56496 C3P0JR 10750186 Ki = 4500 nM T56496 CZ32AV 10784360 Ki = 110 nM T56496 C26QGF 11196556 Ki = 1400 nM T56496 C1N3XD 11208994 Ki = 170 nM T56496 CNR9T0 11209657 Ki = 230 nM T56496 CPDB85 11222591 Ki = 1300 nM T56496 CSO14D 11222628 Ki = 93000 nM T56496 CW61GQ 11232465 Ki = 190 nM T56496 CB60EC 11235364 Ki = 88000 nM T56496 CY5PN7 11244672 Ki = 5100 nM T56496 C5S4XJ 11245059 Ki = 36000 nM T56496 CDL73Y 11257061 Ki = 250000 nM T56496 CT7RW5 11303206 Ki = 40000 nM T56496 CQS04K 11312887 Ki = 750 nM T56496 CD7QH1 11313333 Ki = 23 nM T56496 CMC5T1 11325218 Ki = 28 nM T56496 C5F8OZ 11325652 Ki = 2600 nM T56496 CO7YZ8 11326749 Ki = 9200 nM T56496 CP0VD1 11337570 Ki = 1.8 nM T56496 C1DQB8 11348278 Ki = 18000 nM T56496 C3MFA0 11349134 Ki = 66000 nM T56496 C59XSF 11349331 Ki = 33000 nM T56496 CT2K7O 11349402 Ki = 99 nM T56496 C9ZH7X 11349774 Ki = 1.4 nM T56496 CCJ4Q2 11360541 Ki = 7700 nM T56496 CNKE94 11394776 Ki = 17 nM T56496 C9MN8G 11438678 Ki = 790 nM T56496 CD2K3P 11439655 Ki = 890000 nM T56496 C2DRX9 11450547 Ki = 3400 nM T56496 C57FQS 11460195 Ki = 72 nM T56496 CHX1W8 11484843 Ki = 11000 nM T56496 CZ0U7E 11485425 Ki = 610 nM T56496 C4WP7K 11500379 Ki = 94 nM T56496 C3KGH4 11501582 Ki = 5300 nM T56496 CXO38S 11501635 Ki = 900 nM T56496 CD1U8R 11514463 Ki = 680 nM T56496 CUT09K 11514913 Ki = 6000 nM T56496 CDU57R 11522432 Ki = 200 nM T56496 C0M5KT 11531025 Ki = 250 nM T56496 CFD6R0 11546250 Ki = 37000 nM T56496 C0QR6O 11558328 Ki = 3100 nM T56496 CTL6G5 11566070 Ki = 3200 nM T56496 C5AU3X 11566312 Ki = 2100 nM T56496 C5EJU6 11582118 Ki = 110000 nM T56496 CU9BL8 11597095 Ki = 15000 nM T56496 CJ3O5C 11601371 Ki = 3400 nM T56496 C1JC8F 11608298 Ki = 170 nM T56496 CA25OR 11632695 Ki = 9400 nM T56496 CR0NS3 11639665 Ki = 13000 nM T56496 COYL49 11645402 Ki = 5600 nM T56496 CTCW08 11680583 Ki = 980 nM T56496 C1R7OY 11739550 Ki = 4600 nM T56496 CV8B6A 11772571 Ki = 1200 nM T56496 CV69XM 11772989 Ki = 5900 nM T56496 CZV7K2 11776489 Ki = 4.9 nM T56496 C39PJF 11819842 Ki = 1500 nM T56496 CIW61A 12595069 Ki = 29 nM T56496 CMR38H 12595071 Ki = 30 nM T56496 C6S0UP 12595085 Ki = 59 nM T56496 CPBH15 12595086 Ki = 20 nM T56496 CU8DX7 12595087 Ki = 52 nM T56496 CR6XO1 12606920 Ki = 1.3 nM T56496 C9WV8S 16082606 Ki = 32000 nM T56496 C7SO2P 16082608 Ki = 1300 nM T56496 CV28AH 16082610 Ki = 67000 nM T56496 CKM52A 16082612 Ki = 14000 nM T56496 CUI3A9 16082614 Ki = 2400 nM T56496 CB27SG 16082616 Ki = 18000 nM T56496 C3Q4OY 16082618 Ki = 72000 nM T56496 CY38NR 16082631 Ki = 1400 nM T56496 CICV95 16216219 Ki = 220 nM T56496 CW06SP 18377285 Ki = 25000 nM T56496 CXM85B 18377398 Ki = 100000 nM T56496 C71TOV 20027470 IC50 = 60000 nM T56496 CKS8I9 20065702 Ki = 61000 nM T56496 C9QYR0 20204011 Ki = 10000 nM T56496 C2W8LP 20299667 IC50 = 2000 nM T56496 CFNH96 20299675 IC50 = 2000 nM T56496 C8GTP7 20299685 IC50 = 100 nM T56496 C6L7HG 21393811 IC50 = 2000 nM T56496 C7FZ8G 21539587 Ki = 23000 nM T56496 CMZL78 21584293 Ki = 490 nM T56496 CJD1K4 21584368 Ki = 17 nM T56496 C38LHF 21687108 Ki = 530000 nM T56496 C21YHR 22018495 Ki = 20000 nM T56496 CFJ41D 23336575 Ki = 790 nM T56496 CFX35P 44286717 Ki = 1000 nM T56496 C2HGT1 44287137 Ki = 180000 nM T56496 CE7LR0 44287195 Ki = 12 nM T56496 C0VOW7 44287234 Ki = 13000 nM T56496 CBO94A 44340588 Ki = 41000 nM T56496 CAN1E0 44340624 Ki = 21000 nM T56496 CWU9K6 44363251 Ki = 1200 nM T56496 CDRP38 44363399 Ki = 4400 nM T56496 CJ8NC6 44377597 IC50 = 5000 nM T56496 CLW7K3 44377693 IC50 = 100000 nM T56496 CH4GC6 44377694 IC50 = 2000 nM T56496 CWFR80 44377697 IC50 = 100000 nM T56496 CB2ST0 44377698 IC50 = 50000 nM T56496 CRW5Z8 44377699 IC50 = 7000 nM T56496 CA47OV 44377707 IC50 = 300 nM T56496 C2P9TY 44392584 Ki = 510 nM T56496 C7KD0E 44392595 Ki = 350 nM T56496 CS1ZV6 44392609 Ki = 1400 nM T56496 C92VUC 44392613 Ki = 1700 nM T56496 CJ8NA9 44405400 Ki = 1900 nM T56496 C2P7TG 44405404 Ki = 990 nM T56496 CNM71F 44405405 Ki = 460 nM T56496 CLGE30 44405406 Ki = 4200 nM T56496 CY9BL5 44405407 Ki = 1900 nM T56496 CT1C2F 44405440 Ki = 500 nM T56496 C4YUS1 44405471 Ki = 60000 nM T56496 C0QHU8 44405493 Ki = 1900 nM T56496 CFH35N 44405494 Ki = 8000 nM T56496 C9V1NR 44405495 Ki = 17 nM T56496 C4AXG5 44405498 Ki = 480 nM T56496 CA3IP7 44405499 Ki = 4400 nM T56496 CLJI95 44405506 Ki = 940 nM T56496 CQJ26O 44405513 Ki = 4600 nM T56496 C5CQ9L 44428299 Ki = 900 nM T56496 C7P6CT 44428300 Ki = 33000 nM T56496 C90KAR 44428301 Ki = 2100 nM T56496 CE43QV 44428302 Ki = 910 nM T56496 C6QG9I 44428303 Ki = 2300 nM T56496 CSI52O 44447164 Ki = 5800 nM T56496 C5J0BO 44447165 Ki = 40000 nM T56496 C2T1IS 44447166 Ki = 1200 nM T56496 C5IUT1 44447167 Ki = 2600 nM T56496 C0XH1G 44447169 Ki = 15000 nM T56496 CWSP27 44447170 Ki = 730 nM T56496 C18HWC 44447171 Ki = 21000 nM T56496 CTR97I 44447172 Ki = 9600 nM T56496 CP2K7C 44447173 Ki = 480 nM T56496 CFK9B2 44447174 Ki = 150000 nM T56496 C3IHJ0 44447176 Ki = 3300 nM T56496 CAU72I 44447180 Ki = 17000 nM T56496 C27WNX 44590556 Ki = 40 nM T56496 C0CLD3 54770687 IC50 = 80 nM T56496 CIES80 54771594 IC50 = 10000 nM T56496 CP0FS5 54771824 IC50 = 1000 nM T56496 CW0C4P 155517779 IC50 > 100000 nM T56496 D01SRL 6424833 Ki = 120 nM T56496 D01SRS 15407445 Ki = 72 nM T56496 D03EPY 7046 Ki = 5800 nM T56496 D05ZKW 121938 Ki = 10 nM T56496 D06CMJ 3127 IC50 = 300000 nM T56496 D0C9DC 123920 Ki = 1.55 nM T56496 D0E8HU 10654599 Ki = 820 nM T56496 D0H1WR 5226 Ki = 120 nM T62553 C0N8AB 512986 IC50 = 36000 nM T62553 C0PB1Y 512989 IC50 = 860 nM T62553 CN1R9O 512990 IC50 = 880 nM T62553 CD20ZM 512991 IC50 = 24 nM T62553 C3GU9T 515251 IC50 = 15 nM T62553 CIJC18 515252 IC50 = 435 nM T62553 C6YP3L 515253 IC50 = 42000 nM T62553 CK58FD 515254 IC50 = 7 nM T62553 CO45XM 515255 IC50 = 3 nM T62553 CBO59N 515256 IC50 = 140 nM T62553 CXP13E 515257 IC50 = 635 nM T62553 C9EU0J 515258 IC50 = 5 nM T62553 CO24PB 515259 IC50 = 670 nM T62553 CD4P2V 515260 IC50 = 240 nM T62553 CEB7U2 515261 IC50 = 800 nM T62553 CFSO67 515263 IC50 = 3000 nM T62553 C9B3NT 515264 IC50 = 10 nM T62553 C0OF9T 515340 IC50 = 60000 nM T62553 CH2C5Y 515343 IC50 = 36000 nM T62553 CU7JI4 5274912 IC50 = 20000 nM T62553 C3JK9S 5274914 IC50 = 60000 nM T62553 CQ49CO 5274916 IC50 = 60000 nM T62553 CHDY42 5274917 IC50 = 150000 nM T62553 C5G3UN 5274918 IC50 = 60000 nM T62553 C9YK4Z 5274920 IC50 = 40000 nM T62553 C8RK5X 5274923 IC50 = 60000 nM T62553 CRX6E5 5478832 IC50 = 36000 nM T62553 C4D2IJ 5478833 IC50 = 36000 nM T62553 C4LPJ3 6320476 IC50 = 190000 nM T62553 C79RCS 6320477 IC50 = 60000 nM T62553 C86HJX 6320478 IC50 = 60000 nM T62553 CY01TF 6320479 IC50 = 60000 nM T62553 CJ73SA 6320481 IC50 = 55000 nM T62553 C6T9RU 6320482 IC50 = 323000 nM T62553 CY93NU 6320485 IC50 = 55000 nM T62553 CVG9O1 6320489 IC50 = 48000 nM T62553 CS3N7Y 6320490 IC50 = 68000 nM T62553 C9GB2I 10507528 IC50 = 750000 nM T62553 C07MSU 10626863 IC50 = 100000 nM T62553 C5ZVE0 10675092 IC50 = 35 nM T62553 CG4CE5 10697784 IC50 = 110000 nM T62553 C2EU3H 14517919 IC50 = 60000 nM T62553 C40UGO 14520657 IC50 = 55000 nM T62553 C0GO2C 14520668 IC50 = 60000 nM T62553 C7U4NP 14520672 IC50 = 60000 nM T62553 CR0SL5 14520674 IC50 = 55000 nM T62553 C8H2YC 14520688 IC50 = 400000 nM T62553 C47VOD 14520694 IC50 = 44000 nM T62553 CAMY92 14520700 IC50 = 55000 nM T62553 CEF5G0 15611605 IC50 = 60000 nM T62553 CQ2K8B 15611607 IC50 = 50000 nM T62553 CO5X8J 44376222 IC50 = 12000 nM T62553 C3GQ1N 44376675 IC50 = 44000 nM T62553 C2T4JG 44376943 IC50 = 60000 nM T62553 CB4O3H 56675162 IC50 = 15000 nM T62553 CC87NO 73345557 IC50 = 15000 nM T62553 C9M2PS 73350164 IC50 = 33000 nM T62553 C5BW1C 73353133 IC50 = 29000 nM T62553 CW1O0R 73353134 IC50 = 13000 nM T62553 CL5XS8 73353135 IC50 = 36000 nM T62553 CGS7T1 73354470 IC50 = 108 nM T62553 C7AC0N 73354654 IC50 = 42000 nM T62553 C1QSH7 73356031 IC50 = 41000 nM T87166 D0C6MS 46181428 EC50 = 90 nM T87166 D0E3TC 44259 IC50 = 0.81 nM T87166 D0M5PH 46916694 EC50 = 174 nM T87166 D0O8BS 16039797 EC50 = 28 nM T87166 C9IS6E 449003 EC50 = 67.11 nM T87166 CJL96W 647685 EC50 = 2511.89 nM T87166 C7S0WO 847246 EC50 > 30000 nM T87166 C1TH0W 1172823 EC50 > 100000 nM T87166 C69THW 1445399 EC50 > 100000 nM T87166 CVE10B 2092675 EC50 = 800 nM T87166 CT38DU 2831706 EC50 = 10000 nM T87166 CNCX30 9799942 EC50 = 26700 nM T87166 CF3V5J 9819610 EC50 = 140 nM T87166 C9SR0F 9868203 EC50 = 130 nM T87166 CO3DZ4 9886086 EC50 = 334 nM T87166 C73TXE 9934507 EC50 = 3200 nM T87166 CJ6C5Z 9954194 EC50 = 90 nM T87166 CZ5OM8 10004541 EC50 = 60 nM T87166 C5UPD0 10073655 EC50 = 2600 nM T87166 C6AYU9 10095113 EC50 = 250 nM T87166 CQY6H0 10161315 EC50 = 400 nM T87166 CL4H5Q 10250045 EC50 = 3470 nM T87166 C7F3HR 10252364 EC50 = 200 nM T87166 CN2BH8 10342654 EC50 = 76 nM T87166 C4AJ5Q 10344232 EC50 = 110 nM T87166 C9NAM2 10365275 EC50 = 27.7 nM T87166 C2SX5F 10366412 EC50 = 70 nM T87166 C6L5FA 10385853 EC50 = 2300 nM T87166 CNZ9O8 10408333 EC50 = 1690 nM T87166 C2T9SV 10411846 EC50 = 250 nM T87166 CMYX47 10412882 EC50 = 160 nM T87166 CO8LM0 10432843 EC50 = 57 nM T87166 CL2M1C 10448235 EC50 = 10770 nM T87166 C4HM3V 10454363 EC50 = 38 nM T87166 CH67IC 10455369 EC50 = 40 nM T87166 C5M9FS 10458369 EC50 = 120 nM T87166 CNG18C 10476292 EC50 = 130 nM T87166 CFQ7Z9 10478302 EC50 = 89 nM T87166 C7GRV6 11154711 EC50 = 60 nM T87166 C1QWM8 11178027 EC50 = 110 nM T87166 CA5F2P 11179025 EC50 = 1100 nM T87166 CSYH81 11188508 EC50 = 210 nM T87166 C5LU7E 11235541 EC50 = 160 nM T87166 CA56HS 11270610 EC50 = 180 nM T87166 C8CS5F 11282651 EC50 = 60 nM T87166 CAU59O 11294219 EC50 = 70 nM T87166 CT4HL6 11340230 EC50 = 30 nM T87166 CJB10C 11340776 EC50 = 30 nM T87166 CWS1K4 11363673 EC50 = 40 nM T87166 C2GBC0 11409307 EC50 = 70 nM T87166 CZ2NE9 11476499 EC50 = 60 nM T87166 C4N1CF 11477557 EC50 = 50 nM T87166 C7H9AB 11495849 EC50 = 40 nM T87166 CY4KA2 11501028 EC50 = 210 nM T87166 CIJ51X 11539903 EC50 = 61 nM T87166 CC9OT4 11562233 EC50 = 40 nM T87166 CFC7D3 11576079 EC50 = 32 nM T87166 CQY6U2 11589677 EC50 = 40 nM T87166 C3V9LT 11604824 EC50 = 16.2 nM T87166 CUPN65 11605090 EC50 = 70 nM T87166 C5ZLH8 11610032 EC50 = 60 nM T87166 CZ4B9T 11612643 EC50 = 110 nM T87166 C6EGB7 11626833 EC50 = 31 nM T87166 CD83GL 11634069 EC50 = 37 nM T87166 CO68YB 11634336 EC50 = 73 nM T87166 CWHK19 11641315 EC50 = 35 nM T87166 CEBF28 11647637 EC50 = 80 nM T87166 CQR2N9 11649204 EC50 = 90 nM T87166 CF92JA 11660390 EC50 = 920 nM T87166 CXPC31 11662060 EC50 = 53 nM T87166 CI54QB 11662332 EC50 = 50 nM T87166 CFG52E 11690454 EC50 = 30 nM T87166 CTZ61B 11704809 EC50 = 50 nM T87166 C1QM0R 11711284 EC50 = 70 nM T87166 CXK45U 11718171 EC50 = 80 nM T87166 CGL8A5 11741138 EC50 = 560 nM T87166 CE3ZP2 11743862 EC50 = 37 nM T87166 CFC0X5 11751490 EC50 = 90 nM T87166 CI0YQ1 11752100 EC50 = 30 nM T87166 CHFW18 15942650 EC50 = 70 nM T87166 C8AB4L 16039796 EC50 = 60 nM T87166 CXQ0H2 16039798 EC50 = 370 nM T87166 CA7QW1 16039834 EC50 = 36 nM T87166 CEAW60 16061466 EC50 = 687 nM T87166 CSF6K5 16071499 EC50 = 170 nM T87166 CQ06FD 16071731 EC50 = 47 nM T87166 CLDN06 16349380 EC50 > 100000 nM T87166 CM3Q4D 16660015 EC50 = 4940 nM T87166 C39QRJ 16660016 EC50 = 12300 nM T87166 CRGN27 16660017 EC50 = 7780 nM T87166 CU57HQ 16660167 EC50 = 1700 nM T87166 CFR63A 16660168 EC50 = 3220 nM T87166 CI87GN 16660170 EC50 = 796 nM T87166 CSW71Y 16660174 EC50 = 235 nM T87166 CKVG75 16660331 EC50 = 3440 nM T87166 C47XYC 16660507 EC50 = 77 nM T87166 CB4XC2 16660671 EC50 = 231 nM T87166 C35CLN 16660844 EC50 = 356 nM T87166 C7QG8I 16660845 EC50 = 240 nM T87166 CX2Q9F 16770707 EC50 = 2600 nM T87166 C1C6IQ 20119064 EC50 > 30000 nM T87166 C18QVO 20119572 EC50 = 1400 nM T87166 CC3A0I 23067400 EC50 = 130 nM T87166 CV8NT7 23067404 EC50 = 540 nM T87166 CDT42X 23067415 EC50 = 120 nM T87166 C57YFE 23067440 EC50 = 400 nM T87166 C69YFJ 23067445 EC50 = 180 nM T87166 CHR19Q 23092601 EC50 = 120 nM T87166 CANG15 23092965 EC50 = 210 nM T87166 C2G9VI 23093036 EC50 = 240 nM T87166 C8G2JF 23093050 EC50 = 70 nM T87166 CFJ6M1 23093081 EC50 = 200 nM T87166 CZA86C 23145121 EC50 = 1900 nM T87166 CAJ6W4 23145122 EC50 = 1500 nM T87166 C43PXU 23145136 EC50 = 2700 nM T87166 CSV40P 23145223 EC50 = 5470 nM T87166 C7WP8E 23145280 EC50 = 6100 nM T87166 C1TFP3 23145371 EC50 > 30000 nM T87166 CH5K0X 23145414 EC50 = 1900 nM T87166 CLYF58 23145444 EC50 = 1600 nM T87166 CV7W8N 23145448 EC50 = 7400 nM T87166 C5VC3D 23145556 EC50 = 19100 nM T87166 CK4S1H 23145594 EC50 = 1100 nM T87166 C8BQX5 23145643 EC50 = 630 nM T87166 CVG3S6 23145787 EC50 = 1900 nM T87166 C9IO7D 23160260 EC50 = 570 nM T87166 C5LMT3 23160263 EC50 = 150 nM T87166 CT5GQ2 23160266 EC50 = 30 nM T87166 CC6L9X 23160272 EC50 = 110 nM T87166 CZ2BJ0 23160279 EC50 = 800 nM T87166 CEX53L 23160285 EC50 = 950 nM T87166 C1ZKM8 23160287 EC50 = 40 nM T87166 C3EA6V 23160298 EC50 = 240 nM T87166 C7ETG3 23160304 EC50 = 2700 nM T87166 CY0AN2 23160316 EC50 = 40 nM T87166 CSEG32 23160348 EC50 = 10 nM T87166 CF0J9G 24745013 EC50 = 50000 nM T87166 CX0TY5 24745328 EC50 = 10000 nM T87166 C8WF7O 24745820 EC50 = 2000 nM T87166 CUQ96E 24768019 EC50 = 26 nM T87166 C3Q5VI 24906074 EC50 > 10000 nM T87166 C2DNP8 24906075 EC50 = 580 nM T87166 CK14VC 24906076 EC50 = 140 nM T87166 C8CNK3 24906118 EC50 = 1430 nM T87166 CSQR46 24906119 EC50 = 570 nM T87166 CD3X7A 24906120 EC50 = 70 nM T87166 C1WG4Y 24962524 EC50 = 1600 nM T87166 C8VR6J 24962881 EC50 = 200 nM T87166 C14LMA 24962885 EC50 = 1600 nM T87166 CQJI78 24971095 EC50 = 88 nM T87166 CYB7M8 25069589 EC50 = 400 nM T87166 C7X5FO 25070876 EC50 = 1000 nM T87166 C57WVG 25071203 EC50 = 310 nM T87166 CM16RG 25072138 EC50 = 250 nM T87166 C84TXY 25073999 EC50 = 200 nM T87166 CO4VQ3 25229552 EC50 = 330 nM T87166 CH42VW 25235801 EC50 = 9.5 nM T87166 CV61FP 44224002 EC50 = 122 nM T87166 C35ELW 44224189 EC50 = 3500 nM T87166 CI75AC 44224190 EC50 = 910 nM T87166 CN3I1D 44263455 EC50 = 12560 nM T87166 CCG4S6 44263463 EC50 = 1870 nM T87166 CI85RN 44263467 EC50 = 2530 nM T87166 C5JOR9 44263472 EC50 = 2130 nM T87166 CL8M2J 44263477 EC50 = 1360 nM T87166 CRV3U9 44400835 EC50 > 10000 nM T87166 C8G3AK 44400862 EC50 > 10000 nM T87166 CO6D1U 44400874 EC50 > 10000 nM T87166 CS0XJ7 44400943 EC50 = 650 nM T87166 CKW9S3 44400984 EC50 > 10000 nM T87166 CR63ND 44401001 EC50 = 910 nM T87166 CTR97J 44401059 EC50 = 420 nM T87166 C4UOJ3 44401073 EC50 = 100 nM T87166 C63KDE 44401138 EC50 = 1260 nM T87166 C3M8GL 44401270 EC50 = 130 nM T87166 C92PJC 44401271 EC50 = 4220 nM T87166 C5QRI4 44401302 EC50 = 90 nM T87166 CY0N7T 44401351 EC50 > 10000 nM T87166 CGE9F8 44401406 EC50 > 10000 nM T87166 CT3O4N 44401426 EC50 = 290 nM T87166 CMRZ87 44401503 EC50 = 1780 nM T87166 C6W9IO 44401535 EC50 = 170 nM T87166 CAZ50E 44401560 EC50 > 10000 nM T87166 CF6DK5 44402618 EC50 = 1330 nM T87166 COE69F 44410834 EC50 = 110 nM T87166 C9LYA0 44410892 EC50 = 950 nM T87166 C30KMJ 44410893 EC50 = 610 nM T87166 C0R5NI 44410896 EC50 = 5510 nM T87166 C5FV6R 44410908 EC50 = 20 nM T87166 CAZT49 44410910 EC50 = 90 nM T87166 CE1JU2 44513475 EC50 > 100000 nM T87166 C7HSB1 44513802 EC50 = 7900 nM T87166 CA0D9B 44555462 EC50 = 60 nM T87166 C3PDO9 44564889 EC50 = 1700 nM T87166 CJNC38 44564932 EC50 = 100 nM T87166 C45ZGK 44564933 EC50 = 140 nM T87166 CN7V8U 44564986 EC50 = 200 nM T87166 CBD41N 44564987 EC50 = 220 nM T87166 CLU90G 44564988 EC50 = 380 nM T87166 CD35YR 44564989 EC50 = 100 nM T87166 CL40YN 44565039 EC50 = 120 nM T87166 C6X9UZ 44565040 EC50 = 180 nM T87166 C1TD0Z 44565041 EC50 = 230 nM T87166 C5B9RG 44565042 EC50 > 10000 nM T87166 CWO36Y 44565084 EC50 > 10000 nM T87166 CMI2R3 44565085 EC50 > 10000 nM T87166 C2DTO6 44565086 EC50 = 130 nM T87166 CQY1U5 44565087 EC50 = 110 nM T87166 CRJH83 44565088 EC50 = 420 nM T87166 CGK20W 44565089 EC50 = 420 nM T87166 CUTX37 44565138 EC50 = 930 nM T87166 CG7E9X 44565139 EC50 > 10000 nM T87166 CSNC29 44568124 EC50 = 26010 nM T87166 C1N4TF 44572162 EC50 = 450 nM T87166 CXIC74 44572202 EC50 = 2200 nM T87166 CXSV07 44572245 EC50 = 4200 nM T87166 CD0N7T 44572246 EC50 = 820 nM T87166 CK94TP 44572247 EC50 = 2300 nM T87166 CY8H3I 44572248 EC50 = 5900 nM T87166 CH5KC4 44572249 EC50 = 1100 nM T87166 C47SLQ 44572250 EC50 = 1100 nM T87166 CO9UA5 44572296 EC50 = 3400 nM T87166 C6HVK1 44572297 EC50 = 490 nM T87166 C7ZU9B 44572298 EC50 = 1900 nM T87166 CGI1M2 44572299 EC50 > 30000 nM T87166 C8JA9X 44572300 EC50 > 30000 nM T87166 CLRJ36 44572358 EC50 = 1900 nM T87166 CGW0M3 44572359 EC50 = 2100 nM T87166 CV7D0L 44572360 EC50 = 440 nM T87166 C82QJR 44572361 EC50 = 610 nM T87166 COT3I4 44572411 EC50 = 940 nM T87166 C8CJ1F 44572412 EC50 = 350 nM T87166 CXA70N 44572413 EC50 = 90 nM T87166 C7ZOP2 44593462 EC50 = 1500 nM T87166 CN7I9A 44598465 EC50 = 360 nM T87166 C0LRQ2 45101475 EC50 = 49 nM T87166 C67UVW 45267160 EC50 = 160 nM T87166 CUDS17 45267214 EC50 > 30000 nM T87166 CW3VX8 45267725 EC50 = 930 nM T87166 CB73UE 45268085 EC50 = 90 nM T87166 C1H6LP 45268088 EC50 = 4200 nM T87166 C9MN3O 45268959 EC50 = 240 nM T87166 C9T1LI 45268965 EC50 > 30000 nM T87166 CF24NQ 45269441 EC50 > 30000 nM T87166 CO8X5L 45269804 EC50 = 7400 nM T87166 CRL5E4 45269808 EC50 = 60 nM T87166 CW5T7V 45269833 EC50 = 1600 nM T87166 C30GUD 45270565 EC50 = 970 nM T87166 CWD3K1 45270633 EC50 = 120 nM T87166 C8DTY5 45270647 EC50 = 300 nM T87166 C0LX5E 45270655 EC50 = 910 nM T87166 C1B9VL 45271116 EC50 = 2400 nM T87166 CYB35A 45271117 EC50 = 1700 nM T87166 C74LFZ 45271402 EC50 = 100 nM T87166 C2OL8Y 45271457 EC50 = 110 nM T87166 CL2K5R 45271479 EC50 = 1200 nM T87166 C9KL5V 45271999 EC50 = 1100 nM T87166 CQ35JW 45272000 EC50 = 3000 nM T87166 CCL7V2 45272367 EC50 = 7300 nM T87166 CQX16O 45272819 EC50 > 30000 nM T87166 C9D3QR 45272825 EC50 = 9600 nM T87166 CW6G5U 45272843 EC50 = 1500 nM T87166 CA0SG5 45273147 EC50 = 120 nM T87166 CWEH57 45273248 EC50 = 50 nM T87166 CNMC35 45483579 EC50 = 20 nM T87166 C0MDQ8 45483589 EC50 = 4000 nM T87166 CI7GU2 45483594 EC50 = 200 nM T87166 CG83BX 45483603 EC50 = 40 nM T87166 C8B4MK 45483611 EC50 = 40 nM T87166 CHB1V8 45483612 EC50 = 180 nM T87166 C3QC6O 45483613 EC50 = 80 nM T87166 CB2P1J 45483614 EC50 = 50 nM T87166 CLK12Q 45483615 EC50 = 100 nM T87166 CBW72E 45483616 EC50 = 40 nM T87166 C32YDN 46175430 EC50 = 316.23 nM T87166 CH5Y4W 46175432 EC50 = 398.11 nM T87166 C6MI2B 46175433 EC50 = 78 nM T87166 CZ8SI1 46175518 EC50 = 125.89 nM T87166 CR9J1S 46175520 EC50 = 96 nM T87166 CZKB10 46175521 EC50 = 63.1 nM T87166 CA6G8I 46175610 EC50 = 199.53 nM T87166 C2L3HT 46175611 EC50 = 78 nM T87166 C2Z7LU 46181350 EC50 = 201 nM T87166 C5RAO8 46181353 EC50 = 114 nM T87166 CY6LB8 46181505 EC50 > 10000 nM T87166 CE3P0M 46181581 EC50 = 1080 nM T87166 CLXP57 46181585 EC50 = 2490 nM T87166 CG63YR 46181586 EC50 > 10000 nM T87166 CQYW63 46181666 EC50 = 565 nM T87166 C7XD9Y 46181668 EC50 = 456 nM T87166 CZV05G 46194692 EC50 = 2860 nM T87166 C3MTW9 46194694 EC50 = 2930 nM T87166 CEO0Y4 46194695 EC50 = 1350 nM T87166 CE0XG7 46194836 EC50 = 1040 nM T87166 CO0FM2 46194837 EC50 = 310 nM T87166 CCZ20X 46194838 EC50 = 1000 nM T87166 C3BOA6 46194839 EC50 = 355 nM T87166 CA82KH 46194840 EC50 = 724 nM T87166 CDF0L5 46194841 EC50 = 1180 nM T87166 C47CTV 46195120 EC50 = 26 nM T87166 CO7T2E 46226664 EC50 = 70 nM T87166 CM8GY3 46226671 EC50 = 220 nM T87166 CLZ5A6 46226674 EC50 = 120 nM T87166 C4LH0C 46226682 EC50 > 5000 nM T87166 CISU59 46226685 EC50 = 60 nM T87166 C82ADZ 46226690 EC50 = 120 nM T87166 CU25HV 46226704 EC50 = 80 nM T87166 CPF46K 46226705 EC50 > 5000 nM T87166 C14CRW 46226729 EC50 = 110 nM T87166 C2ISV8 46226734 EC50 = 100 nM T87166 CIT94H 46844903 EC50 = 158 nM T87166 CCIW59 46907147 EC50 = 330 nM T87166 C2S4MO 46907148 EC50 = 157 nM T87166 CYXP74 46907180 EC50 = 320 nM T87166 C49TVJ 46907261 EC50 = 61 nM T87166 CI9MJ3 46907262 EC50 = 120 nM T87166 CBO85R 46907263 EC50 = 79 nM T87166 C1SZR4 46907264 EC50 = 2860 nM T87166 C65YKG 46909841 EC50 = 990 nM T87166 CHQ51D 46910963 EC50 = 1930 nM T87166 CAZT21 46911020 EC50 = 980 nM T87166 C07MBF 46911021 EC50 = 510 nM T87166 CV5WQ3 46911072 EC50 = 910 nM T87166 CI6VA9 46911123 EC50 = 230 nM T87166 C1MEW3 46911124 EC50 = 114 nM T87166 CA30VH 46911180 EC50 = 391 nM T87166 CAYT85 46911181 EC50 = 770 nM T87166 C2UQ7T 46916741 EC50 = 210 nM T87166 CI8DX5 53629543 EC50 = 52 nM T87166 C7C4UK 54580432 EC50 = 230 nM T87166 C7W6IK 54580433 EC50 = 60 nM T87166 C2IEY4 54580434 EC50 = 260 nM T87166 C15JOP 54580435 EC50 = 140 nM T87166 CC5F3J 54580718 EC50 > 10000 nM T87166 C04BQW 54581442 EC50 = 560 nM T87166 C6MY8W 54581443 EC50 = 330 nM T87166 CPGZ47 54581444 EC50 = 700 nM T87166 C9OPY8 54581445 EC50 = 1300 nM T87166 CF38PO 54581717 EC50 = 60 nM T87166 CZ4S3E 54582448 EC50 = 440 nM T87166 C8W1TB 54582449 EC50 = 670 nM T87166 CC14SQ 54582450 EC50 = 160 nM T87166 CZD53X 54582451 EC50 = 1500 nM T87166 C4GY6Z 54582452 EC50 = 720 nM T87166 CI08VJ 54583427 EC50 = 160 nM T87166 CSAW51 54583428 EC50 = 1300 nM T87166 CT69ZN 54583686 EC50 = 90 nM T87166 CCBN26 54584389 EC50 = 500 nM T87166 C24UVI 54584390 EC50 = 110 nM T87166 CA4WS9 54584391 EC50 = 70 nM T87166 C2C7HZ 54584650 EC50 = 100 nM T87166 C1S7RY 54584651 EC50 = 40 nM T87166 CB73KV 54585342 EC50 = 510 nM T87166 CPVA60 54585344 EC50 = 240 nM T87166 CQSD21 54585345 EC50 = 600 nM T87166 C65APY 54585346 EC50 = 590 nM T87166 C7C6TJ 54585347 EC50 = 260 nM T87166 CP8T5E 54585589 EC50 = 110 nM T87166 C0DZS3 54585590 EC50 = 400 nM T87166 CBAW81 54586307 EC50 = 66 nM T87166 CG7QV6 54586308 EC50 = 3300 nM T87166 CAY91M 54587333 EC50 = 480 nM T87166 C0R8KP 54587334 EC50 = 1500 nM T87166 C2Y0VQ 54587595 EC50 > 10000 nM T87166 CVE1U6 54587596 EC50 = 100 nM T87166 CB6S2N 54765712 EC50 = 90 nM T87166 CBER71 54765716 EC50 = 110 nM T87166 CC0GM3 54765880 EC50 = 1100 nM T87166 C64PDY 54766044 EC50 = 590 nM T87166 CSL5Y9 54766195 EC50 = 200 nM T87166 CWPX40 54766199 EC50 = 440 nM T87166 CE38ZA 54766497 EC50 = 1000 nM T87166 CI4B1H 54766500 EC50 = 230 nM T87166 C9QYW8 54767116 EC50 = 200 nM T87166 C53KCX 54767117 EC50 = 830 nM T87166 C1MU0C 54767118 EC50 = 70 nM T87166 CT5N1Q 54767119 EC50 = 7500 nM T87166 C0USC9 54767120 EC50 = 940 nM T87166 CLW86X 54767447 EC50 = 150 nM T87166 CTD03G 54767610 EC50 = 850 nM T87166 C8M5XN 54767782 EC50 = 500 nM T87166 CIK06P 54767784 EC50 = 1400 nM T87166 C9E5CN 54767786 EC50 = 230 nM T87166 CPR46H 54767787 EC50 = 170 nM T87166 CJOS85 56640458 EC50 = 330 nM T87166 CXD19C 56640459 EC50 = 350 nM T87166 C3FSE8 56640460 EC50 = 450 nM T87166 C2Y9PW 56640461 EC50 = 180 nM T87166 CCK56W 56640462 EC50 > 20000 nM T87166 C19RXG 56640529 EC50 = 300 nM T87166 C8C6JF 56640530 EC50 = 640 nM T87166 C3MQ0J 56640532 EC50 = 1350 nM T87166 CHBX89 56640533 EC50 = 290 nM T87166 C4JPG9 56640596 EC50 = 170 nM T87166 CQ5UM1 56640597 EC50 > 20000 nM T87166 CYK3S9 56640598 EC50 = 210 nM T87166 CL35SI 56640599 EC50 = 790 nM T87166 C3WB8U 56645356 IC50 > 20000 nM T87166 CC1ZG8 56832521 IC50 = 1420 nM T87166 C8K6XM 56955210 EC50 > 10000 nM T87166 CO3H7M 56955211 EC50 > 10000 nM T87166 CZ1L2E 56955212 EC50 = 284 nM T87166 CJX75E 56968094 EC50 = 80 nM T87166 CHO7W4 57461474 EC50 = 630 nM T87166 CS3EB8 57461532 EC50 = 120 nM T87166 CWA9F6 57482815 EC50 > 100000 nM T87166 C2QS1Y 57504248 EC50 = 316.23 nM T87166 C6ESZ4 57504261 EC50 = 316.23 nM T87166 CNAJ67 57504264 EC50 = 100 nM T87166 CMB2W7 57504266 EC50 = 50.12 nM T87166 CAY71X 57504268 EC50 = 125.89 nM T87166 C70HUQ 57504283 EC50 = 630.96 nM T87166 C02DMC 57504292 EC50 = 3162.28 nM T87166 C9ZA6Y 57504293 EC50 = 794.33 nM T87166 CBU6N2 57504311 EC50 = 1584.89 nM T87166 C6S8CV 57504312 EC50 = 5011.87 nM T87166 C0W5QD 57504313 EC50 = 158.49 nM T87166 CD85MW 57504320 EC50 = 125.89 nM T87166 CH79YV 57504325 EC50 = 158.49 nM T87166 CZ8SF5 57504326 EC50 = 251.19 nM T87166 CRC5O1 57504327 EC50 = 1258.93 nM T87166 C7JDH2 57504328 EC50 = 501.19 nM T87166 CM8Z6N 57504345 EC50 = 199.53 nM T87166 CKE12J 57504346 EC50 = 316.23 nM T87166 C4UAZ5 57504347 EC50 = 125.89 nM T87166 CH3Y9K 57504348 EC50 = 125.89 nM T87166 C9TY4W 57504354 EC50 = 630.96 nM T87166 CCT08G 57504355 EC50 = 630.96 nM T87166 C0OIW2 57504356 EC50 = 501.19 nM T87166 CPQA09 57504358 EC50 = 316.23 nM T87166 CP7BL3 57504360 EC50 = 398.11 nM T87166 CV20RS 57504361 EC50 = 630.96 nM T87166 C42OWY 57504362 EC50 = 501.19 nM T87166 C8K7TB 57504363 EC50 = 501.19 nM T87166 C7X5KI 57504373 EC50 = 199.53 nM T87166 CPR02A 57504388 EC50 = 1584.89 nM T87166 CI74AT 57504389 EC50 = 501.19 nM T87166 COB73U 57504402 EC50 = 199.53 nM T87166 CLWU10 57504418 EC50 = 630.96 nM T87166 C8UHW1 57504419 EC50 = 794.33 nM T87166 C0BGQ4 57504420 EC50 = 2511.89 nM T87166 C38YSV 57504421 EC50 = 3162.28 nM T87166 C1CPF8 57504444 EC50 = 79.43 nM T87166 CB54GY 57504445 EC50 = 199.53 nM T87166 CYHT79 57504446 EC50 = 501.19 nM T87166 CAV2N7 57504447 EC50 = 199.53 nM T87166 C3AOX7 57504450 EC50 = 50.12 nM T87166 CR0HE5 57504454 EC50 = 251.19 nM T87166 CV8B0T 57504457 EC50 = 501.19 nM T87166 CRLJ46 57504462 EC50 = 316.23 nM T87166 CNEB25 57504463 EC50 = 199.53 nM T87166 CR1A8Z 57504467 EC50 = 630.96 nM T87166 CP8O6G 57504472 EC50 = 199.53 nM T87166 C9EIU6 57504473 EC50 = 100 nM T87166 C90OLN 57504474 EC50 = 63.1 nM T87166 C4SXY9 57657277 EC50 = 200 nM T87166 C7TRJ8 57657292 EC50 = 250 nM T87166 C38DEZ 57657324 EC50 = 63 nM T87166 CEC68K 57665301 EC50 = 6300 nM T87166 C7NLM4 57665307 EC50 = 790 nM T87166 C0AW4L 57665314 EC50 = 1200 nM T87166 C9SIC2 57665343 EC50 = 160 nM T87166 CURL06 57665404 EC50 = 630 nM T87166 C49AVI 57963961 EC50 = 500 nM T87166 C6LX7O 57963993 EC50 = 120 nM T87166 CAO7L3 57963994 EC50 = 630 nM T87166 CRP2S7 57964003 EC50 > 100000 nM T87166 C1RH9X 57964005 EC50 = 630 nM T87166 C9CQ1S 57964007 EC50 = 790 nM T87166 CWHF76 57964017 EC50 = 120 nM T87166 C05TAW 57964021 EC50 = 31 nM T87166 C18HQO 57964044 EC50 = 2000 nM T87166 CX6Z7H 57964096 EC50 = 4000 nM T87166 CZ1Y2I 57964111 EC50 = 100 nM T87166 CGL3E7 57964129 EC50 = 40 nM T87166 CFEG70 58967446 EC50 = 7900 nM T87166 C5Y9UO 59225642 EC50 = 325 nM T87166 C4H5QL 59225645 EC50 = 208 nM T87166 C2GZ9X 59225669 EC50 = 2640 nM T87166 C53HDO 59279483 EC50 = 125.89 nM T87166 CN1Y9X 59279548 EC50 = 158.49 nM T87166 CC1AN4 59279550 EC50 = 79.43 nM T87166 CM4XB0 59279551 EC50 = 158.49 nM T87166 CMLX58 59483313 EC50 = 153 nM T87166 CK26YS 59560375 EC50 = 9.4 nM T87166 C2UAL6 60150713 EC50 = 44.8 nM T87166 C5P9BI 60150714 EC50 = 28.3 nM T87166 CW71YI 66582327 IC50 = 524 nM T87166 C07OER 66582448 IC50 = 9 nM T87166 C59AVC 66582451 IC50 = 343 nM T87166 CXY93Z 66582550 IC50 = 6 nM T87166 C1V4AM 66582747 EC50 > 50000 nM T87166 CZP63S 66582940 IC50 = 90 nM T87166 C3J4PB 66583294 IC50 = 7 nM T87166 C78SJP 67305655 EC50 = 135 nM T87166 C04DLF 67305810 EC50 = 216 nM T87166 CWSR01 67306982 EC50 = 184 nM T87166 CN4PR7 67307127 EC50 = 217 nM T87166 CM0L1P 67996575 EC50 = 7500 nM T87166 C2IXM6 67996937 EC50 = 9200 nM T87166 C1QI6T 70654666 EC50 = 1200 nM T87166 C7W8DN 70655077 IC50 = 16 nM T87166 C0IHR4 70655459 IC50 = 25 nM T87166 C6X1TV 70655709 IC50 = 56 nM T87166 C0GZ2U 70655743 IC50 = 14 nM T87166 CWJK41 70681373 EC50 = 62.6 nM T87166 CYMW45 70681393 EC50 = 78 nM T87166 CGH6P2 70681394 EC50 = 90.1 nM T87166 CHID07 70681408 EC50 = 491 nM T87166 C1U6IP 70683468 EC50 = 48 nM T87166 CL0NY6 70683488 EC50 = 165 nM T87166 CQ74MO 70683489 EC50 > 1000 nM T87166 CFDJ76 70685511 EC50 = 360 nM T87166 CH7X5V 70685578 EC50 = 47.7 nM T87166 COK4Y3 70685590 EC50 = 65.4 nM T87166 CNM4V3 70685591 EC50 = 52.3 nM T87166 CGB89C 70685618 EC50 = 144 nM T87166 C2S5PZ 70685619 EC50 = 63.1 nM T87166 C58DNJ 70685620 EC50 = 460 nM T87166 CWK02C 70687665 EC50 = 60 nM T87166 CG80EM 70687724 EC50 = 52 nM T87166 CXBA02 70687742 EC50 = 250 nM T87166 CML2A8 70689789 EC50 = 90.4 nM T87166 CCG18H 70689790 EC50 = 297 nM T87166 C8U1JR 70689814 EC50 = 242 nM T87166 CV7Z8R 70691929 EC50 = 890 nM T87166 CTM81Y 70691949 EC50 = 265 nM T87166 CQDY31 70691950 EC50 = 83.5 nM T87166 C4W0SE 70693981 EC50 = 95.1 nM T87166 CQ5DI8 70694001 EC50 = 44.8 nM T87166 CW5S4U 70696106 EC50 = 101 nM T87166 C9KCJ1 70696107 EC50 = 64.6 nM T87166 CV42XS 71295771 EC50 = 4000 nM T87166 COIL91 71295772 EC50 = 3100 nM T87166 C14OWJ 71450444 EC50 = 2320 nM T87166 CL3FD1 71450445 EC50 = 1540 nM T87166 C6V8UB 71450638 EC50 > 100000 nM T87166 CX7J5R 71454074 EC50 = 620 nM T87166 CZU43H 71454075 EC50 = 710 nM T87166 CV2P8F 71454226 EC50 > 100000 nM T87166 CDW0Y8 71454227 EC50 = 15848.93 nM T87166 C6B3US 71455985 EC50 = 501.19 nM T87166 COL05V 71457592 EC50 = 440 nM T87166 C6TU7Y 71457593 EC50 = 880 nM T87166 C30PNK 71459489 EC50 = 310 nM T87166 CRFV16 71461227 EC50 = 340 nM T87166 C6P2TR 71461228 EC50 = 2030 nM T87166 CHY12O 71463148 EC50 = 1584.89 nM T87166 C9K4PJ 71533605 EC50 = 70 nM T87166 CB7CR8 71540507 EC50 = 283 nM T87166 CHO86E 71540508 EC50 = 239 nM T87166 C3U8IF 71540509 EC50 = 852 nM T87166 CV6XY7 71540510 EC50 = 80 nM T87166 C9JOI1 71540511 EC50 = 119 nM T87166 CX9PQ7 71540610 EC50 = 109 nM T87166 CW40NO 71540611 EC50 = 200 nM T87166 CEQ48V 71540612 EC50 = 161 nM T87166 CC6V5S 71540613 EC50 = 848 nM T87166 CXC3G5 71540614 EC50 = 115 nM T87166 C1N4AU 71540615 EC50 = 132 nM T87166 CS3TY9 71540726 EC50 = 131 nM T87166 C7W3RT 71540727 EC50 = 855 nM T87166 C32CJR 71540841 EC50 = 296 nM T87166 CLU18T 71540842 EC50 = 165 nM T87166 CG4MR5 71540843 EC50 = 284 nM T87166 C6MR9G 71540844 EC50 = 56 nM T87166 COS46D 71540845 EC50 = 120 nM T87166 CFR68W 71540962 EC50 = 95 nM T87166 CE2JW7 71540963 EC50 = 134 nM T87166 C8HYV5 71540964 EC50 = 90 nM T87166 CTM10G 71540965 EC50 = 778 nM T87166 C9QB2W 71540966 EC50 = 83 nM T87166 C4UXN2 71579462 EC50 > 100000 nM T87166 CZ5JI1 71579463 EC50 > 100000 nM T87166 C3JOX6 71579464 EC50 = 4000 nM T87166 CGI8P2 71579465 EC50 > 100000 nM T87166 CTYQ32 71579556 EC50 = 1000 nM T87166 CG15IO 71579557 EC50 = 2000 nM T87166 C30HZK 71579558 EC50 = 10000 nM T87166 C84BIF 71579559 EC50 = 500 nM T87166 CIC8E0 71579643 EC50 = 1200 nM T87166 C4ZL6I 71579644 EC50 = 2500 nM T87166 CVU9S7 71579645 EC50 = 79 nM T87166 CMY31V 71579646 EC50 = 310 nM T87166 C5OP6T 71579738 EC50 = 400 nM T87166 C6A9WI 71579739 EC50 = 630 nM T87166 CWA2Y0 71579740 EC50 = 5000 nM T87166 CD9CL2 71579741 EC50 = 2000 nM T87166 C6T7WH 71579742 EC50 = 1600 nM T87166 CY90QZ 71579834 EC50 = 790 nM T87166 CCZI90 71579835 EC50 = 2000 nM T87166 CQ1X6I 71579836 EC50 = 160 nM T87166 CPU96R 71579931 EC50 = 2000 nM T87166 C0RVW5 71579932 EC50 = 79 nM T87166 CCJ6U7 71579933 EC50 = 1000 nM T87166 C5R6FI 71579934 EC50 = 160 nM T87166 CB5OV7 71580026 EC50 = 500 nM T87166 CFX48K 71580027 EC50 = 1200 nM T87166 CVC6K8 71603520 EC50 = 160 nM T87166 CJG4A1 71603523 EC50 = 72 nM T87166 CGI54Z 71603582 EC50 = 130 nM T87166 CS1KL2 71603583 EC50 = 130 nM T87166 CZ72JT 71603584 EC50 = 350 nM T87166 C6HRO9 71603585 EC50 = 60 nM T87166 CO3X7L 71627422 EC50 = 2000 nM T87166 CXO3Z7 71715871 IC50 = 56 nM T87166 CCB2T3 71715872 IC50 = 1430 nM T87166 C06OGC 71813336 EC50 = 740 nM T87166 CIY5E7 71813504 EC50 > 100000 nM T87166 CFI6O3 71813669 EC50 = 23000 nM T87166 C20AID 71814304 EC50 = 3800 nM T87166 CM87ET 72703061 EC50 = 119 nM T87166 C3QEY8 72705641 EC50 = 562 nM T87166 CABU30 72723937 EC50 = 137 nM T87166 C8QZ1U 72723938 EC50 = 113 nM T87166 C27JGL 72724082 EC50 = 227 nM T87166 CWLO53 72724083 EC50 = 1350 nM T87166 CV35EN 72724084 EC50 > 10000 nM T87166 C7MO0V 73053709 IC50 = 4 nM T87166 CLA35R 73332001 IC50 = 5 nM T87166 CTUE84 73350645 EC50 = 110 nM T87166 C1CXY7 73659150 IC50 = 87 nM T87166 C0Q7UT 76310478 IC50 = 439 nM T87166 C3EWZ2 76310479 IC50 = 26 nM T87166 CM3B1F 76310480 IC50 = 1010 nM T87166 C2DTJ9 76314132 IC50 = 44 nM T87166 C7V1KW 76314133 IC50 = 324 nM T87166 C29PEI 76314158 IC50 = 6 nM T87166 CC6H2P 76317706 IC50 = 2 nM T87166 C81KJP 76317707 IC50 = 252 nM T87166 CY9HK6 76321415 IC50 = 645 nM T87166 C81FAI 76321432 IC50 = 484 nM T87166 C1SNL7 76325010 IC50 = 445 nM T87166 CXM72J 76328584 IC50 = 316 nM T87166 C0TN1H 76328603 IC50 = 779 nM T87166 C71IUO 76332259 IC50 = 8630 nM T87166 CRQ28W 76335899 IC50 = 484 nM T87166 CD2Q8U 76685070 EC50 = 6 nM T87166 CIK9R7 76685222 EC50 = 95 nM T87166 CX2ZD0 76900521 EC50 = 9.6 nM T87166 C1M3WD 76902401 EC50 = 51.5 nM T87166 CYQ06P 76902786 EC50 = 14 nM T87166 CD6Z7U 76902970 EC50 = 5.7 nM T87166 CB0HQ7 76902972 EC50 = 68.5 nM T87166 CK4Z0Y 76902974 EC50 = 49 nM T87166 C1T2XV 77050669 EC50 = 0.8 nM T87166 CMT61E 77105088 EC50 > 50000 nM T87166 CSC2Y3 77105090 EC50 = 212 nM T87166 CC9FY4 77105092 EC50 = 7460 nM T87166 C31UXO 77105468 EC50 > 50000 nM T87166 CRI9Z8 77107273 EC50 = 315 nM T87166 CTQ39O 77107274 EC50 > 50000 nM T87166 CP63SW 77107471 EC50 > 50000 nM T87166 CH4OP6 77107475 EC50 = 238 nM T87166 CGD6H2 77107671 EC50 = 807 nM T87166 CP64YI 77107672 EC50 = 441 nM T87166 C71HOU 77460994 EC50 = 280 nM T87166 CI5VR6 78319009 EC50 = 27 nM T87166 CSY95P 78319067 EC50 = 34 nM T87166 CKC7B8 78319068 EC50 = 6 nM T87166 C9Q6LF 78350461 EC50 = 88 nM T87166 C2Q5LG 87420181 EC50 = 100 nM T87166 CBO71W 90253114 EC50 = 3.4 nM T87166 CX2ZC5 90655313 EC50 = 103 nM T87166 CN3UT5 90655314 EC50 = 5 nM T87166 C04PFY 90655315 EC50 > 50000 nM T87166 CYJ2H4 90655316 EC50 = 688 nM T87166 CL2R0E 90655317 EC50 = 2430 nM T87166 CSJ3R1 90655318 EC50 = 8 nM T87166 CDTB80 90655319 EC50 = 33 nM T87166 C7DW0Y 90655320 EC50 = 463 nM T87166 C49SGT 90655321 EC50 = 106 nM T87166 CNU52W 90665343 EC50 = 70 nM T87166 CEST68 90665736 EC50 = 6610 nM T87166 C71ARQ 90665737 EC50 = 870 nM T87166 CZOW03 90665738 EC50 = 3061 nM T87166 CVJE69 90665739 EC50 = 92 nM T87166 CHO63U 90665740 EC50 = 480 nM T87166 C58VON 90665741 EC50 > 20 nM T87166 C9EXG1 90665742 EC50 > 5000 nM T87166 CPD02Y 90665743 EC50 = 85 nM T87166 CT65NK 90665744 EC50 = 64 nM T87166 CJC4T0 90665745 EC50 = 261 nM T87166 CUD10X 90665746 EC50 = 393 nM T87166 CQ9E2Z 90665747 EC50 = 705 nM T87166 CKFN19 90665748 EC50 > 5000 nM T87166 C0DQN8 90665749 EC50 > 5000 nM T87166 C4WK9H 90665750 EC50 = 2170 nM T87166 CJ2D3R 90665751 EC50 = 477 nM T87166 CR62PM 90665752 EC50 = 391 nM T87166 CJX07M 90665753 EC50 = 127 nM T87166 C62TXE 90665754 EC50 = 167 nM T87166 CH91MY 90665755 EC50 = 254 nM T87166 CMSC59 90665756 EC50 = 331 nM T87166 CPV6M0 90665757 EC50 > 100000 nM T87166 C4JH3B 90665883 EC50 = 520 nM T87166 CA2HQ5 90665884 EC50 = 1800 nM T87166 CVT7D0 90665885 EC50 = 1440 nM T87166 CKT31A 90665886 EC50 = 11350 nM T87166 CV87YZ 90665887 EC50 = 1520 nM T87166 C5I0ZO 90665888 EC50 > 20000 nM T87166 CWE2M0 90665889 EC50 = 220 nM T87166 CU9MV6 90666148 EC50 = 73 nM T87166 CIM1S7 90667868 EC50 = 316.23 nM T87166 CKE53T 118709612 IC50 = 176 nM T87166 CW6ZS2 118709613 IC50 = 201 nM T87166 C1VF6C 118709614 IC50 = 112 nM T87166 CM16RA 118709615 IC50 = 1110 nM T87166 C0BZL9 118709616 IC50 = 601 nM T87166 CAYD23 118709617 IC50 = 33 nM T87166 CX14CU 118709618 IC50 = 14 nM T87166 C10YGB 118709619 IC50 = 5 nM T87166 CX6K8P 118709620 IC50 = 49 nM T87166 CWS9N0 118709621 IC50 = 17 nM T87166 C1PKC3 118709622 IC50 = 201 nM T87166 CG19YT 118709623 IC50 = 1 nM T87166 CS59BP 118709624 IC50 = 5 nM T87166 CYFZ80 118709625 IC50 = 23 nM T87166 CE5OJ3 118709626 IC50 = 87 nM T87166 C4BS3V 118709627 IC50 = 40 nM T87166 C0K8CS 118709628 IC50 = 30000 nM T87166 CLI39N 118709629 IC50 = 19 nM T87166 C3FK2T 118709630 IC50 = 5 nM T87166 C9V6TN 118709631 IC50 = 7 nM T87166 CF65MN 118709632 IC50 = 7 nM T87166 CH1P0O 118709633 IC50 = 8 nM T87166 C9D8KO 118709634 IC50 = 11 nM T87166 C4KQ5Z 118709635 IC50 = 6 nM T87166 CD86MA 118709636 IC50 = 309 nM T87166 C0EMB7 118709637 IC50 = 50 nM T87166 CQMG41 118709638 IC50 = 42 nM T87166 CA4XE7 118709639 IC50 = 21 nM T87166 CL85ET 118709640 IC50 = 24 nM T87166 CBI5D2 118709641 IC50 = 11 nM T87166 CF8AS5 118709642 IC50 = 29 nM T87166 CTR72O 118709643 IC50 = 40 nM T87166 CADG08 118709644 IC50 = 16 nM T87166 CYUQ39 118709645 IC50 = 17 nM T87166 CP6XL9 118709646 IC50 = 47 nM T87166 C6ODH8 118709647 IC50 = 35 nM T87166 C6NK0I 118709648 IC50 = 20 nM T87166 C4QZ1U 118709649 IC50 = 15 nM T87166 CGH14P 118709650 IC50 = 20 nM T87166 CO2J3B 118709651 IC50 = 33 nM T87166 CH7M0E 118709652 IC50 = 60 nM T87166 CWS2I6 118709653 IC50 = 1950 nM T87166 C0DK6P 118709654 IC50 = 27 nM T87166 CW0O8P 118709655 IC50 = 48 nM T87166 CKW1S8 118715090 EC50 = 13200 nM T87166 C4JEV2 118715091 EC50 > 50000 nM T87166 CHOT73 118715092 EC50 > 50000 nM T87166 C8QO5T 118715093 EC50 = 203 nM T87166 CSDT09 118715094 EC50 = 1730 nM T87166 CH9D3E 118715095 EC50 > 50000 nM T87166 CUYS91 118715096 EC50 = 2120 nM T87166 CNR7J3 118715097 EC50 = 1620 nM T87166 CB3O7Q 118715098 EC50 = 758 nM T87166 CD5W4F 118715099 EC50 = 952 nM T87166 CVM0P1 118715100 EC50 = 393 nM T87166 C56LKZ 118715101 EC50 = 276 nM T87166 CX5J2W 118715102 EC50 = 172 nM T87166 C1NB5T 118715103 EC50 = 262 nM T87166 CKSJ32 118715104 EC50 = 319 nM T87166 CFB3J6 118715105 EC50 = 345 nM T87166 CI84SB 118715106 EC50 = 3093 nM T87166 C89GKF 118715107 EC50 = 172 nM T87166 CYT6Q2 118715108 EC50 = 550 nM T87166 C4J1LO 118715109 EC50 = 182 nM T87166 CXJ21M 118715110 EC50 = 317 nM T87166 CMDT90 118715126 EC50 = 233 nM T87166 C7LR6D 118715127 EC50 = 132 nM T87166 CQEC09 118715128 EC50 = 111 nM T87166 CWU61I 118715129 EC50 = 195 nM T87166 CMC42V 118722859 EC50 = 120 nM T87166 CCX5G8 118722860 EC50 = 590 nM T87166 C3UCB1 118722861 EC50 = 440 nM T87166 C3HL7T 118722862 EC50 = 110 nM T87166 CD6NA4 118722863 EC50 = 1590 nM T87166 C7RG1C 118722864 EC50 = 350 nM T87166 C0FTA8 118722865 EC50 = 110 nM T87166 CZE2I8 118722866 EC50 = 14 nM T87166 CUH56Q 118722867 EC50 = 290 nM T87166 CU1R7X 118722868 EC50 = 460 nM T87166 C4MZ5H 118722869 EC50 = 370 nM T87166 CFE76U 118722870 EC50 = 16800 nM T87166 C4Z7OI 118722871 EC50 = 7980 nM T87166 CQ8O9D 118722872 EC50 = 490 nM T87166 C0N8QF 118722873 EC50 = 350 nM T87166 COK7P2 118722874 EC50 = 2760 nM T87166 CMYE62 118722875 EC50 = 820 nM T87166 C2MX7J 118722876 EC50 = 68 nM T87166 CZGB41 118722877 EC50 = 97 nM T87166 COJ5M6 118723158 EC50 = 500 nM T87166 CX7N9L 122177975 EC50 = 1870 nM T87166 CLF06W 122177976 EC50 = 7700 nM T87166 CK87HG 122177977 EC50 = 301 nM T87166 CK60NM 122177978 EC50 = 25 nM T87166 CU34FI 122177979 EC50 = 21 nM T87166 C5KF2R 122177980 EC50 = 12 nM T87166 CK4U0A 122177981 EC50 = 30 nM T87166 CJ17UX 122177982 EC50 = 39 nM T87166 CP3Q4Y 122177983 EC50 = 37 nM T87166 CL5O3I 122177984 EC50 = 163 nM T87166 CF1SM2 122177985 EC50 = 6 nM T87166 CIM8X1 122177986 EC50 = 6 nM T87166 CC2Z8V 122177987 EC50 = 20 nM T87166 CIC09Q 122177988 EC50 = 39 nM T87166 CH8YJ0 122177989 EC50 = 9 nM T87166 CKM9N7 122177990 EC50 = 53 nM T87166 CSYT18 122177991 EC50 = 46 nM T87166 C3MWQ0 122177992 EC50 = 6 nM T87166 CRQU30 122177993 EC50 = 7 nM T87166 CSW58B 122177994 EC50 = 16 nM T87166 C29PFM 122178417 EC50 = 121 nM T87166 C1K3WT 122178418 EC50 = 24 nM T87166 CJI3Z2 122178419 EC50 = 191 nM T87166 CU31IB 122417289 EC50 = 5420 nM T87166 CF69NM 122417290 EC50 = 150 nM T87166 CQB0A3 122417291 EC50 = 90 nM T87166 C1ZMV5 122417292 EC50 > 10000 nM T87166 C13LAU 122417306 EC50 > 10000 nM T87166 CNT36W 122417307 EC50 > 10000 nM T87166 CQ3ON6 122417309 EC50 = 7080 nM T87166 CGRD78 122417311 EC50 = 100 nM T87166 C1ON9E 122417314 EC50 = 8420 nM T87166 CCV0U1 122417331 EC50 > 10000 nM T87166 CQ89PN 122417334 EC50 = 2220 nM T87166 C7L1FJ 122417335 EC50 = 870 nM T87166 CW49RO 122417336 EC50 = 890 nM T87166 CFOS92 122417341 EC50 = 210 nM T87166 C6QB1C 122417381 EC50 = 820 nM T87166 CO1BV3 122417386 EC50 = 30 nM T87166 C5V0WS 122417387 EC50 = 1090 nM T87166 CSGA91 127037884 EC50 = 1260 nM T87166 CYIA64 127038219 EC50 = 2930 nM T87166 C27YQS 127038882 EC50 = 38300 nM T87166 CJTB32 127039203 EC50 = 255 nM T87166 CE01UJ 127039539 EC50 = 263 nM T87166 C9F8KT 127040025 EC50 = 783 nM T87166 C98LOI 127040026 EC50 = 756 nM T87166 CVJ38E 127040028 EC50 = 1410 nM T87166 C59KQR 127040029 EC50 = 810 nM T87166 CF1O0U 127040030 EC50 = 2050 nM T87166 C4Z5FC 127040362 EC50 = 194 nM T87166 C5WVX6 127041333 EC50 = 1240 nM T87166 C72FSB 127041335 EC50 = 688 nM T87166 CU1D5W 127041336 EC50 = 342 nM T87166 C7Z0QB 127041338 EC50 = 608 nM T87166 C2IE9J 127041529 EC50 = 6630 nM T87166 CNU46R 127041530 EC50 = 1870 nM T87166 C2H8NB 127041532 EC50 = 1300 nM T87166 CN5L1G 127041828 EC50 = 535 nM T87166 CF6V7W 127042444 EC50 = 173 nM T87166 CAH79D 127042445 EC50 = 638 nM T87166 C4B3RU 127042446 EC50 = 1100 nM T87166 CO2B6Z 127042447 EC50 = 3290 nM T87166 CC9BK1 127042493 EC50 = 1100 nM T87166 C56ZYK 127042495 EC50 = 12.4 nM T87166 CH7W9L 127042498 EC50 = 115 nM T87166 CVP3F0 127042499 EC50 = 695 nM T87166 C7XO1N 127042500 EC50 = 148 nM T87166 C16QBR 127052916 IC50 = 3500 nM T87166 CGX1L3 136017450 EC50 = 100 nM T87166 C43TFK 136239454 EC50 = 10300 nM T87166 CXEO53 137632657 EC50 = 4.8 nM T87166 C40XJY 137632890 EC50 = 2.1 nM T87166 CA5E1U 137634006 EC50 > 100000 nM T87166 CJ2YR1 137638835 EC50 = 1600 nM T87166 CPY3L1 137640045 EC50 = 3100 nM T87166 CH0IM8 137641773 EC50 = 1 nM T87166 CO0LK7 137642011 EC50 = 1.4 nM T87166 CGXN24 137642601 EC50 = 200 nM T87166 C1XA5R 137645312 EC50 = 1000 nM T87166 CYX97Q 137646747 EC50 < 0.85 nM T87166 CD5U2Y 137646945 EC50 = 5000 nM T87166 CH1TK9 137648705 EC50 = 100 nM T87166 CBA4F8 137650798 EC50 = 4.2 nM T87166 CQCI85 137655205 EC50 = 9.6 nM T87166 CC26QP 141451166 IC50 > 20000 nM T87166 C0Q2WJ 141451172 IC50 > 20000 nM T87166 C1FJ8M 141451182 IC50 > 20000 nM T87166 CV3K0N 145120681 EC50 = 320 nM T87166 C5O9KR 145120691 EC50 = 200 nM T87166 C8MFL2 145120693 EC50 = 170 nM T87166 CO1I7R 145120712 EC50 = 230 nM T87166 C15ETP 145120713 EC50 = 900 nM T87166 C7ZC2T 145120718 EC50 = 180 nM T87166 CM87UG 145120731 EC50 = 140 nM T87166 C3J6RX 145120732 EC50 = 550 nM T87166 C0BJP4 145964031 EC50 = 490 nM T87166 CKW96H 145964360 EC50 = 1130 nM T87166 CFE8C1 145964383 EC50 = 500 nM T87166 CG09UN 145965258 EC50 = 2230 nM T87166 CBP57Z 145965347 EC50 = 290 nM T87166 CV1L9C 145966971 EC50 = 1300 nM T87166 CM4FT2 145967041 EC50 = 170 nM T87166 CAU0J4 145971883 EC50 = 690 nM T87166 CNY7S5 145973008 EC50 = 2600 nM T87166 CBUD81 145973011 EC50 = 7000 nM T87166 CY1T5D 145974954 EC50 = 6080 nM T87166 C2K9OV 145975820 EC50 > 10000 nM T87166 CQ5XK1 145975880 EC50 = 460 nM T87166 CE3SM6 145976246 EC50 = 200 nM T87166 C7V9TB 145976429 EC50 = 230 nM T87166 C9D8SV 145977527 EC50 = 50 nM T87166 CEZF41 145977772 EC50 > 10000 nM T87166 C16USM 145978148 EC50 = 4600 nM T87166 CA1I6B 145978251 EC50 = 210 nM T87166 CS3Q0D 145978396 EC50 = 330 nM T87166 C6NS9M 145978500 EC50 = 300 nM T87166 CSTL91 150436720 EC50 = 880 nM T87166 C6YLC7 150575761 EC50 = 50 nM T87166 C4W3YI 151355906 EC50 = 670 nM T87166 C5TL2E 155511256 EC50 = 190 nM T87166 C2Q4TS 155511463 EC50 = 10800 nM T87166 C80URT 155511835 EC50 > 50000 nM T87166 CJ6HF5 155512123 EC50 = 2130 nM T87166 C2MD1Q 155513187 IC50 > 10000 nM T87166 CP40AV 155514513 EC50 = 310 nM T87166 CE6ZW3 155515486 EC50 = 110 nM T87166 CY3W9U 155517272 EC50 = 6250 nM T87166 CAH7J0 155518537 EC50 = 50 nM T87166 CU5T8M 155522427 EC50 = 66 nM T87166 CZVX84 155522913 EC50 = 120 nM T87166 CF13SN 155525686 EC50 = 170 nM T87166 C4MS8I 155532809 EC50 = 230 nM T87166 CQ0P4I 155533510 EC50 = 830 nM T87166 CAP54S 155533635 IC50 > 20000 nM T87166 CP64OM 155533971 EC50 = 47 nM T87166 CLZ95T 155534084 EC50 = 920 nM T87166 C2UQS8 155535024 EC50 = 120 nM T87166 C6A5VU 155535512 EC50 = 97 nM T87166 CV1AE4 155538180 IC50 > 20000 nM T87166 CB9DU3 155539930 EC50 = 110 nM T87166 C0IBP2 155540236 EC50 = 66 nM T87166 CAOQ49 155541450 EC50 = 36 nM T87166 C2X9BV 155543626 EC50 = 98 nM T87166 C7T0HB 155543920 EC50 = 290 nM T87166 CAB9J3 155544468 EC50 = 88 nM T87166 C7Z0TH 155544957 EC50 = 14 nM T87166 C90EDX 155545320 EC50 = 37 nM T87166 CN6V3Z 155545330 EC50 = 2300 nM T87166 CGK09E 155545349 EC50 = 6700 nM T87166 CH92MR 155545937 EC50 = 40 nM T87166 CZ23XT 155545997 EC50 = 45 nM T87166 C8S7KU 155547616 EC50 = 110 nM T87166 CZ9WB3 155548914 EC50 = 300 nM T87166 C6HZV2 155550743 EC50 = 130 nM T87166 CVKS30 155555013 EC50 = 45 nM T87166 CUBW79 155556274 EC50 = 72 nM T87166 C5KP4J 155557173 IC50 > 20000 nM T87166 CP37KC 155558714 EC50 = 38 nM T87166 CE41AY 155561677 EC50 = 60 nM T87166 CN2YD7 155563130 EC50 = 660 nM T87166 CMC1H5 155563873 EC50 = 40 nM T87166 C6H1GB 155563881 EC50 = 500 nM T87166 C1GSW0 155564114 EC50 = 530 nM T87166 C7U4KI 155568209 EC50 = 160 nM T87166 CHCY62 155568860 EC50 = 83 nM T87166 CWPV14 155568928 EC50 = 51 nM T87166 D02XFR 899301 EC50 = 6300 nM T87166 D04QGH 10432339 EC50 = 364 nM T87166 D0P0PP 10044792 EC50 = 570 nM T33901 D0K0EK 5881 EC50 > 10000 nM T33901 CVEP92 91474 EC50 = 8700 nM T33901 CFA5H9 91498 EC50 = 1700 nM T33901 CCT25S 102008 EC50 = 3400 nM T33901 C6L3XW 159461 EC50 = 1700 nM T33901 CA56RZ 168038 EC50 = 2900 nM T33901 CW95KX 3489642 IC50 = 4400 nM T33901 C0JE4T 4573798 IC50 = 2500 nM T33901 C95KUL 10319758 EC50 = 1500 nM T33901 CUX78W 11101442 EC50 = 4000 nM T33901 CR20DF 14238178 EC50 = 4300 nM T33901 CZ97IL 15251407 EC50 = 3400 nM T33901 CV57AQ 24768125 EC50 = 3100 nM T33901 CMY6Z1 44574013 IC50 = 20 nM T33901 C3X9PI 44574014 IC50 = 660 nM T33901 CK20DH 44574015 IC50 = 7400 nM T33901 CM2H7J 44574016 IC50 = 79000 nM T33901 CM0EC5 44574038 IC50 = 81000 nM T33901 CA4TH0 44574039 IC50 = 4600 nM T33901 CLV5D4 44574063 IC50 = 390 nM T33901 CNR2F3 53316716 IC50 = 4800 nM T33901 C1PV5U 53316749 IC50 = 6100 nM T33901 C6XW5O 53316750 IC50 = 8200 nM T33901 C4PF0R 53316751 IC50 = 4200 nM T33901 C2IYH0 53316752 IC50 = 3300 nM T33901 CL4GO0 53317350 IC50 = 4200 nM T33901 CV8O9R 53317351 IC50 = 4600 nM T33901 CB3Z1R 53318010 IC50 = 8300 nM T33901 CF35ZE 53318044 IC50 = 1100 nM T33901 C48RZD 53318045 IC50 = 2600 nM T33901 CY02QK 53318046 IC50 = 4700 nM T33901 CPK4N2 53318047 IC50 = 16900 nM T33901 C8E2MR 53318048 IC50 = 3100 nM T33901 C24BIP 53318629 IC50 = 14500 nM T33901 C4UJE7 53318630 IC50 = 5500 nM T33901 CF01VD 53318631 IC50 = 3100 nM T33901 C1SC0M 53318966 IC50 = 3200 nM T33901 C8H2GZ 53319044 IC50 = 8700 nM T33901 C0T3XL 53319355 IC50 = 16600 nM T33901 C4QWV7 53319357 IC50 = 23600 nM T33901 CSZ1W2 53319358 IC50 = 10900 nM T33901 C2W8JI 53319389 IC50 = 4000 nM T33901 C3GF6I 53319391 IC50 = 4200 nM T33901 C8T1MD 53319953 IC50 = 13700 nM T33901 CJ0L6S 53319954 IC50 = 12900 nM T33901 C28HFC 53319956 IC50 = 10300 nM T33901 CY2ZQ9 53319957 IC50 = 8300 nM T33901 CW3ZI2 53319958 IC50 = 3800 nM T33901 CRU70F 53319959 IC50 = 14200 nM T33901 CDGV95 53320633 IC50 = 11800 nM T33901 CH0S4Q 53320663 IC50 = 9400 nM T33901 CX6I2W 53320664 IC50 = 4600 nM T33901 CAVQ05 53320695 IC50 = 4800 nM T33901 C0YE7H 53320696 IC50 = 9500 nM T33901 C97LBP 53320697 IC50 = 3800 nM T33901 CR6Y5D 53321259 IC50 = 2100 nM T33901 CF1KB7 53321636 IC50 = 3500 nM T33901 CECO67 53321956 IC50 = 6400 nM T33901 C9AUY5 53321989 IC50 = 1100 nM T33901 CSN8M4 53321990 IC50 = 2500 nM T33901 C7QC6G 53322578 IC50 = 5500 nM T33901 CE8Z2A 53322580 IC50 = 1000 nM T33901 C7FB8K 53322581 IC50 = 6500 nM T33901 CH8F9L 53322582 IC50 = 2600 nM T33901 CK0YX2 53322915 IC50 = 19000 nM T33901 C2WQY7 53323307 IC50 = 11400 nM T33901 CHJ6B3 53323308 IC50 = 2500 nM T33901 C83WIM 53323349 IC50 = 3100 nM T33901 CS34NW 53323350 IC50 = 900 nM T33901 CJEM18 53323351 IC50 = 8200 nM T33901 C9GCT2 53323919 IC50 = 4200 nM T33901 C86LDZ 53323920 IC50 = 1700 nM T33901 C6Q5JT 53323921 IC50 = 14000 nM T33901 C2Z7XV 53323922 IC50 = 6000 nM T33901 CY10RT 53323923 IC50 = 22000 nM T33901 CW60QM 53323924 IC50 = 6300 nM T33901 C6TZ5I 53323925 IC50 = 15000 nM T33901 CM1S3J 53323926 IC50 = 12000 nM T33901 C49SJW 53324636 IC50 = 4400 nM T33901 CREQ62 53324637 IC50 = 19200 nM T33901 CJ4I1U 53324638 IC50 = 59000 nM T33901 CC6G7N 53324639 IC50 = 4500 nM T33901 C25TFG 53324640 IC50 = 5400 nM T33901 C4JYH8 53324653 IC50 = 3800 nM T33901 COW43F 53325198 IC50 = 49000 nM T33901 C3DLI2 53325199 IC50 = 26500 nM T33901 CT2CZ0 53325200 IC50 = 7700 nM T33901 CH78KT 53325201 IC50 = 10400 nM T33901 C6O9RZ 53325202 IC50 = 4500 nM T33901 CL2V7T 53325203 IC50 = 3700 nM T33901 CU1BV3 53325204 IC50 = 2500 nM T33901 C3IDE6 53325206 IC50 = 2000 nM T33901 CQ6XS9 53325208 IC50 = 3900 nM T33901 CE6X9L 53325209 IC50 = 3600 nM T33901 C9BU1V 53325606 IC50 = 1000 nM T33901 CK2CV0 53325945 IC50 = 1300 nM T33901 C1LH7N 53325974 IC50 = 12200 nM T33901 C63JAQ 53326491 IC50 = 7000 nM T33901 C8ADT3 53326907 IC50 = 600 nM T33901 C0PZX4 71771041 EC50 = 1700 nM T33901 CIQB17 118169488 IC50 = 20000 nM T33901 CQ3H9M 118169505 IC50 = 46000 nM T33901 C6EKN3 118169520 IC50 = 18000 nM T33901 C4FHB0 118169537 IC50 = 70000 nM T33901 C2I8LT 118707101 EC50 = 1700 nM T33901 CK0V7Q 118707213 EC50 = 9900 nM T33901 C1C9WJ 118707214 EC50 = 1400 nM T33901 CWU1G4 118707215 EC50 = 4800 nM T33901 CQ09TC 118707216 EC50 = 880 nM T33901 CQHU30 118707217 EC50 = 150 nM T33901 CBHR25 118707218 EC50 = 290 nM T33901 CUN51P 118707219 EC50 = 360 nM T33901 C23DZB 118707221 EC50 = 1800 nM T33901 C18NSC 118707222 EC50 = 1000 nM T33901 C1L6SN 118707223 EC50 = 840 nM T33901 CQG67E 118707224 EC50 = 560 nM T33901 CF54ON 118707298 EC50 = 6100 nM T33901 C0A1WQ 118707300 EC50 = 370 nM T33901 C7MF4O 118707301 EC50 = 6800 nM T33901 C27JDE 118707302 EC50 = 360 nM T33901 CM3WS4 118707303 EC50 > 10000 nM T33901 CTZ3K2 118707304 EC50 = 86 nM T33901 CPJ32N 118729152 IC50 = 88000 nM T33901 CANO50 118729153 IC50 = 54000 nM T33901 CJD61N 11342976 IC50 = 4 nM T33901 CE3L2D 45486567 IC50 = 200 nM T33901 D06OVX 65094 EC50 = 3300 nM T33901 D09XJH 9894653 IC50 = 300 nM T33901 D0FB7S 473141 EC50 = 3400 nM T33901 D0L7PI 473142 EC50 = 1900 nM T61243 D00ENY 33032 EC50 = 1180 nM T61243 D0D4OW 57338826 IC50 = 10500 nM T61243 D0U5CS 213056 EC50 > 100000 nM T61243 CB15YI 125799 EC50 > 1000000 nM T61243 CO9KU6 443586 Ki > 1000000 nM T61243 C7OJ4N 1894361 EC50 = 158.49 nM T61243 COJV81 4521898 EC50 > 10000 nM T61243 C05WNA 5310956 Ki = 230000 nM T61243 C3RTI9 6348408 EC50 = 89000 nM T61243 CD68LI 6604795 Ki > 5000000 nM T61243 CV2MX5 8595992 EC50 = 218.78 nM T61243 C9XQK6 10198133 EC50 > 100000 nM T61243 CQ1L0O 10359073 Ki > 300000 nM T61243 CYL91R 10456810 IC50 = 15350 nM T61243 CASI54 11768848 EC50 > 1000000 nM T61243 CSW38G 15420544 EC50 > 10000 nM T61243 CJS57V 16061421 EC50 = 1970000 nM T61243 CG3Q6X 16739372 EC50 > 1000000 nM T61243 C6Q4GL 16747847 EC50 = 602000 nM T61243 CM7JD0 16747848 EC50 = 625000 nM T61243 CWU3X9 16748099 EC50 > 3000000 nM T61243 CS5B7A 18138918 IC50 > 30000 nM T61243 CJR05E 24780088 EC50 = 169000 nM T61243 C5OQ7F 24780092 EC50 > 100000 nM T61243 C7F4YL 24780225 EC50 > 100000 nM T61243 CUS45D 24905703 EC50 > 1000000 nM T61243 C86BUK 24905705 EC50 > 1000000 nM T61243 CNF72Q 44190035 IC50 > 10000 nM T61243 CR1OL6 44328753 IC50 = 9420 nM T61243 CUA80G 44328850 IC50 = 23070 nM T61243 C2SH0O 44329024 IC50 = 67820 nM T61243 CX0Y4F 44329029 IC50 = 7820 nM T61243 C76LOU 44329031 IC50 = 6250 nM T61243 CCV4N5 44329032 IC50 = 7610 nM T61243 CDP86T 44329033 IC50 = 2600 nM T61243 C9V5XC 44329042 IC50 = 19660 nM T61243 CAK39T 44406220 EC50 = 700000 nM T61243 CH9J0V 44406221 EC50 > 1000000 nM T61243 CSD19C 44429217 EC50 > 1000000 nM T61243 CFAM64 45082292 EC50 > 1000000 nM T61243 CC4P3Q 46215704 EC50 = 5200 nM T61243 C31PAF 46700737 EC50 > 10000 nM T61243 CGS4F2 46836713 EC50 > 10000 nM T61243 CKB74O 46918013 EC50 > 1000000 nM T61243 C1VY4Z 46918015 EC50 = 69000 nM T61243 CWE2O4 51033723 IC50 > 10000 nM T61243 CN1HU8 53235518 EC50 > 10000 nM T61243 CY58NO 53240406 IC50 > 12500 nM T61243 CIHC67 54582001 IC50 > 30000 nM T61243 C93KPD 54815068 EC50 = 1584.89 nM T61243 C49IAZ 57765535 EC50 > 100000 nM T61243 C4BZ0U 57765536 EC50 > 100000 nM T61243 C9QDZ0 57765549 EC50 > 100000 nM T61243 CSI9E0 57765613 EC50 > 100000 nM T61243 CBFD61 57765616 EC50 > 100000 nM T61243 CC82HD 57765622 EC50 > 100000 nM T61243 CQ70WE 57765633 EC50 > 100000 nM T61243 CISA81 58058356 EC50 > 100000 nM T61243 CPDW56 58058372 EC50 > 100000 nM T61243 C8N4UB 60096231 EC50 > 25000 nM T61243 CBX67G 67246999 EC50 > 10000 nM T61243 C5K7QG 67974411 EC50 > 10000 nM T61243 CCT07V 68290289 EC50 > 10000 nM T61243 C03JUE 68290572 EC50 > 10000 nM T61243 C4HI0U 70789291 EC50 > 1000000 nM T61243 C2JS0I 71574837 EC50 > 1000000 nM T61243 CV5IT8 71574838 EC50 > 1000000 nM T61243 CL9BJ8 71574839 EC50 > 1000000 nM T61243 CCS4T2 71574840 EC50 > 1000000 nM T61243 CXW8R2 72714783 EC50 > 10000 nM T61243 C0VN8X 92044496 EC50 = 418000 nM T61243 CCP5U2 122195692 EC50 > 10000 nM T61243 CH2AO4 122539788 IC50 > 30000 nM T61243 C2MEI0 124425164 EC50 = 100000 nM T61243 CFC05Q 131954513 EC50 = 650 nM T61243 CX7L4E 134474664 EC50 = 29.2 nM T61243 C9J1ZX 134521675 EC50 = 6.9 nM T61243 CEQ5Y6 134536725 EC50 = 1.205 nM T61243 CS7O0A 137634883 EC50 > 100000 nM T61243 C9H6NY 137639752 EC50 = 62000 nM T61243 CK2W6L 137640190 EC50 > 100000 nM T61243 CAI63F 137642874 EC50 > 100000 nM T61243 C1FCY7 137643759 EC50 = 11600 nM T61243 C9U6EI 137645989 EC50 = 63000 nM T61243 CCW58E 137646034 EC50 > 100000 nM T61243 C3PDO0 137647077 EC50 > 100000 nM T61243 CO9L1G 137650519 EC50 = 51200 nM T61243 CT1M7B 137654697 EC50 = 295000 nM T61243 CMQ61F 137655963 EC50 = 53800 nM T61243 C9C8KU 137661528 EC50 = 39000 nM T61243 CZ6AN1 145422113 EC50 = 1 nM T61243 CWA8H2 145955288 EC50 = 600 nM T61243 C76FVC 155518354 EC50 = 740 nM T61243 C18EFY 155518933 EC50 = 1584.89 nM T61243 C8IFM7 155547657 EC50 = 109.65 nM T61243 D00EPM 73755217 IC50 > 30000 nM T61243 D00NCL 46836562 EC50 > 10000 nM T61243 D01EVA 6278000 Ki > 100000 nM T61243 D04DKM 104766 Ki > 1000000 nM T61243 D04MVR 11530404 IC50 > 10000 nM T61243 D05TFE 5218788 Ki > 100000 nM T61243 D06DUE 40539 EC50 > 1000000 nM T61243 D06PAK 10058694 Ki > 100000 nM T61243 D07GRG 10197984 Ki > 100000 nM T61243 D07PZQ 68841 EC50 < 200000 nM T61243 D09AQK 4545574 EC50 = 48000 nM T61243 D09QUN 58368068 EC50 > 10000 nM T61243 D0DX6U 23725699 IC50 > 10000 nM T61243 D0EK6P 5310984 Ki > 300000 nM T61243 D0IO8J 3025961 Ki > 100000 nM T61243 D0K2XD 53391766 IC50 = 63 nM T61243 D0LC5O 16062593 EC50 >= 30000 nM T61243 D0N2TP 44190040 IC50 > 10000 nM T61243 D0N9UZ 9819927 Ki = 990 nM T61243 D0OV2V 6324634 Ki > 300000 nM T61243 D0P2VP 11708219 EC50 = 700000 nM T61243 D0PN6Z 179394 Ki = 175000 nM T61243 D0Q6VH 5311432 Ki > 100000 nM T61243 D0W3PY 6604820 EC50 = 280000 nM T02719 D00ENY 33032 Ki = 57.54 nM T02719 D0B6RA 9834591 EC50 = 48 nM T02719 D0T3DG 9886034 Ki = 4.5 nM T02719 D01VZE 67705089 Ki = 2.7 nM T02719 D0D4OW 57338826 IC50 = 46.1 nM T02719 D0P4BQ 9857256 Ki > 10000 nM T02719 D0U5CS 213056 EC50 = 24.3 nM T02719 CY3C2X 4408 EC50 = 39000 nM T02719 COJV81 4521898 EC50 > 10000 nM T02719 C05WNA 5310956 Ki = 440 nM T02719 C7J6KQ 6604704 EC50 = 30000 nM T02719 CD68LI 6604795 Ki > 1000000 nM T02719 C9PJQ1 9794208 EC50 = 0.11 nM T02719 CZL1H9 9861792 EC50 > 300000 nM T02719 C31YKH 9885608 EC50 > 12500 nM T02719 C9XQK6 10198133 Ki = 4.7 nM T02719 CX12HM 10330132 Ki = 52000 nM T02719 CMW4B2 10353365 Ki = 0.17 nM T02719 CZ09YG 10358265 IC50 = 8580 nM T02719 CQ1L0O 10359073 Ki = 6100 nM T02719 C2TRI8 10492773 IC50 = 80 nM T02719 CG48QI 10515174 IC50 = 1400 nM T02719 CP0B8Q 10567792 IC50 = 760 nM T02719 C0P9JO 10587622 IC50 = 650 nM T02719 C20AXL 10607617 IC50 = 2500 nM T02719 C06TDU 10688450 IC50 = 170 nM T02719 CD0E3P 10710505 IC50 = 1200 nM T02719 CBQV60 10732318 IC50 = 2800 nM T02719 C6D9IL 10778385 IC50 = 570 nM T02719 CQE5Y9 10783272 IC50 = 280 nM T02719 C4Q3RT 10807972 IC50 = 16 nM T02719 CACY46 10826383 IC50 = 550 nM T02719 C8MOC5 10828532 IC50 = 80 nM T02719 CHZ17V 10852666 IC50 = 470 nM T02719 CDO7A1 10979251 Ki = 138 nM T02719 CJ5B8P 11084869 EC50 = 6.6 nM T02719 CR7BZ3 11220424 EC50 = 4.96 nM T02719 C8LSU6 11275666 EC50 = 24.9 nM T02719 C3D0LM 11298568 Ki = 146 nM T02719 CL1VX3 11310142 Ki = 302 nM T02719 CX2T1N 11344646 EC50 = 34 nM T02719 CA50PD 11481048 Ki > 100000 nM T02719 C6NY5K 11503055 IC50 = 190 nM T02719 CGX8F6 11596869 EC50 > 12500 nM T02719 CASI54 11768848 EC50 > 1000000 nM T02719 CSW38G 15420544 EC50 > 10000 nM T02719 CP9Y7Q 15479143 EC50 = 0.24 nM T02719 CS5B7A 18138918 IC50 > 30000 nM T02719 C5WYI2 21309795 IC50 = 76.1 nM T02719 CB3T7C 24905650 IC50 > 1000000 nM T02719 CNF72Q 44190035 IC50 > 10000 nM T02719 CL13FV 44302605 IC50 > 300000 nM T02719 C03QML 44302608 IC50 = 16100 nM T02719 C2H6QV 44302609 IC50 > 300000 nM T02719 CP1QS5 44302686 IC50 = 40300 nM T02719 CDM1P2 44302819 IC50 > 300000 nM T02719 C34AVQ 44302856 IC50 = 63600 nM T02719 C9Y6QA 44302913 IC50 > 300000 nM T02719 CKL1M8 44302930 IC50 = 166000 nM T02719 C9U0NH 44302931 IC50 > 300000 nM T02719 CD5XY2 44302932 IC50 > 300000 nM T02719 CWV7F0 44322840 Ki = 100 nM T02719 C2SKJ1 44322921 Ki = 2200 nM T02719 CL47OE 44345358 IC50 = 1800 nM T02719 CSZ48I 44345382 IC50 > 10000 nM T02719 CA57SX 44345536 IC50 > 10000 nM T02719 CGNR10 44345546 IC50 > 10000 nM T02719 CDRU87 44348706 IC50 = 210 nM T02719 CSJE56 44348769 IC50 = 260 nM T02719 CUD35Q 44348846 IC50 = 180 nM T02719 C1IHR4 44348859 IC50 = 200 nM T02719 CI06ET 44348911 IC50 = 420 nM T02719 C2O8QK 44348939 IC50 = 160 nM T02719 CM3T1Q 44348993 IC50 = 180 nM T02719 C7P2EA 44361401 Ki = 3 nM T02719 CF0LY9 44361402 Ki > 10000 nM T02719 CIM8S2 44378268 EC50 = 33000 nM T02719 CFAM64 45082292 Ki = 199526.23 nM T02719 C31PAF 46700737 EC50 > 10000 nM T02719 CGS4F2 46836713 EC50 > 10000 nM T02719 CV6F9U 49799828 IC50 > 300000 nM T02719 C0L2SP 51036108 EC50 > 30000 nM T02719 CAU6D5 51036701 EC50 > 30000 nM T02719 CBI3A0 51036916 EC50 > 30000 nM T02719 C3GQ8O 51037131 EC50 > 30000 nM T02719 CN1HU8 53235518 EC50 > 10000 nM T02719 CY58NO 53240406 EC50 = 129 nM T02719 C9ZGL6 53338952 IC50 = 3800 nM T02719 C60LFJ 53393854 IC50 = 2500 nM T02719 C0WY1J 53393859 IC50 > 10000 nM T02719 C1Y9BR 53393868 IC50 = 2041.74 nM T02719 CIHC67 54582001 IC50 > 30000 nM T02719 CJRG27 54761054 EC50 > 30000 nM T02719 CC6HJ9 56587978 IC50 = 5700 nM T02719 CC5EO2 56587980 IC50 > 10000 nM T02719 CJ8OE4 56587985 IC50 = 3235.94 nM T02719 C1VRF2 56587992 IC50 = 5000 nM T02719 CYAQ39 60096178 Ki = 0.47 nM T02719 C38GPO 60096183 EC50 = 7.15 nM T02719 C2NRC3 60096190 EC50 = 2 nM T02719 C63MKC 60096194 EC50 = 356 nM T02719 CMUL95 60096201 EC50 = 0.71 nM T02719 CW32CB 60096204 Ki = 4.34 nM T02719 C8JAU2 60096211 Ki = 177 nM T02719 C5PSF3 60096224 EC50 = 0.17 nM T02719 CXO4R6 60096228 EC50 = 2.12 nM T02719 C8N4UB 60096231 EC50 = 0.47 nM T02719 C9V3NZ 60096236 EC50 = 5.1 nM T02719 C38CBK 60096246 EC50 = 2.44 nM T02719 CN3OV8 60096250 Ki = 2.29 nM T02719 C4PU9N 67056056 EC50 > 30000 nM T02719 CBX67G 67246999 EC50 > 10000 nM T02719 C06MTQ 67705326 IC50 = 38.5 nM T02719 C7MLP4 67705376 IC50 = 14.3 nM T02719 CB16WU 67707808 IC50 = 20.5 nM T02719 C03HIJ 67973779 EC50 = 290 nM T02719 CRS94B 67973913 EC50 = 150 nM T02719 CJ4HA6 67974346 EC50 = 34 nM T02719 C5K7QG 67974411 EC50 = 6760 nM T02719 C75YSP 67974644 EC50 = 74 nM T02719 CCT07V 68290289 IC50 = 290 nM T02719 C03JUE 68290572 IC50 = 630 nM T02719 CZT05A 69929646 EC50 > 30000 nM T02719 CG7F5Z 70051296 IC50 = 3390 nM T02719 CBK2Y6 70051926 EC50 = 15.5 nM T02719 CZ6XT7 70052526 EC50 = 14.2 nM T02719 CJIX85 71131322 EC50 = 27.3 nM T02719 C4JV5H 71135411 Ki = 62.4 nM T02719 CE8L3P 71136640 EC50 = 235 nM T02719 CGH26Q 71136653 Ki = 126 nM T02719 CW04KN 71136654 EC50 = 77.9 nM T02719 CAN01B 71136655 Ki = 157 nM T02719 CHC91O 71137008 Ki = 79 nM T02719 CH0W1O 71137010 Ki = 56.7 nM T02719 CUB8G1 71137011 Ki = 69 nM T02719 CP07IN 71137012 Ki = 58.3 nM T02719 C28ZBK 71137034 Ki = 63.2 nM T02719 C5LC2E 71450430 IC50 > 10000 nM T02719 CNXB36 71476419 Ki = 65.1 nM T02719 CNIW83 71479388 EC50 > 30000 nM T02719 C8U0CT 71681823 EC50 = 12.3 nM T02719 CO5P1V 71681824 EC50 = 57.1 nM T02719 C6EIO9 71681825 EC50 = 23.5 nM T02719 CLH9N3 71681826 Ki = 272 nM T02719 CXW8R2 72714783 EC50 = 3390 nM T02719 C0HF5W 73347368 IC50 = 4200 nM T02719 C3G4HD 86695984 IC50 = 29.6 nM T02719 C3M8QU 89554892 IC50 > 30000 nM T02719 CWZQ47 90098428 EC50 = 30.5 nM T02719 CK53MQ 117972250 EC50 = 890 nM T02719 C8SYH1 121447916 IC50 > 30000 nM T02719 CCP5U2 122195692 EC50 > 10000 nM T02719 CH2AO4 122539788 IC50 > 30000 nM T02719 C9I2BV 127039660 EC50 = 540 nM T02719 CPZ70S 127052897 EC50 > 30000 nM T02719 C38BRY 131801162 EC50 > 10000 nM T02719 CFC05Q 131954513 EC50 > 10000000 nM T02719 CW31CD 134129940 IC50 = 127 nM T02719 CL2UY8 134132133 IC50 = 153 nM T02719 CP8C5N 134137754 IC50 = 54.1 nM T02719 CQT7H6 134138062 IC50 = 1070 nM T02719 CL7G4D 134139744 IC50 = 83.2 nM T02719 C5I6FC 134141510 IC50 = 85 nM T02719 CR4DE8 134144056 IC50 = 239 nM T02719 C5JNX4 134144441 IC50 = 178 nM T02719 CO1H6B 134152341 IC50 = 185 nM T02719 CL72ZY 134154496 IC50 = 145 nM T02719 CB8W0T 134155683 IC50 = 71 nM T02719 C3EGM5 137321168 IC50 > 10000 nM T02719 CR5AB3 137634033 Ki = 281 nM T02719 C5TQS6 137635882 Ki = 757 nM T02719 CBI4Z5 137656301 Ki = 425 nM T02719 CU2I6G 137659992 EC50 = 4.96 nM T02719 C7ECH8 142469540 EC50 < 100 nM T02719 CI60ZB 142469552 EC50 < 100 nM T02719 CM1QH8 142469564 EC50 < 100 nM T02719 CI2MN3 142469580 EC50 < 100 nM T02719 C97XSR 146523789 EC50 < 100 nM T02719 C60JAC 146523794 EC50 < 100 nM T02719 CGO17P 146523813 EC50 <= 100 nM T02719 CJ3H5D 146576905 EC50 <= 100 nM T02719 C18EFY 155518933 EC50 = 630.96 nM T02719 CYXE53 155538270 IC50 > 10000 nM T02719 CMCG93 155539952 IC50 > 30000 nM T02719 CK4XC6 44322529 Ki = 200 nM T02719 D00EPM 73755217 IC50 > 30000 nM T02719 D00NCL 46836562 EC50 > 10000 nM T02719 D04DKM 104766 EC50 = 30000 nM T02719 D05TFE 5218788 Ki > 100000 nM T02719 D06DUE 40539 Ki = 40000 nM T02719 D06PAK 10058694 Ki = 7.6 nM T02719 D06SDD 9837317 EC50 = 2.07 nM T02719 D07GRG 10197984 EC50 = 4.58 nM T02719 D09AQK 4545574 Ki > 200000 nM T02719 D09QUN 58368068 EC50 > 10000 nM T02719 D09UBS 10428048 Ki > 100000 nM T02719 D09YEQ 11158623 IC50 = 270 nM T02719 D0EK6P 5310984 Ki = 410 nM T02719 D0IO8J 3025961 Ki > 100000 nM T02719 D0N0NJ 15508178 IC50 > 300000 nM T02719 D0N2TP 44190040 IC50 > 10000 nM T02719 D0N9UZ 9819927 IC50 = 10 nM T02719 D0OV2V 6324634 Ki = 30000 nM T02719 D0PN6Z 179394 Ki > 1000000 nM T02719 D0Q6VH 5311432 Ki > 100000 nM T02719 D0R0IB 56587994 IC50 = 660 nM T46814 D00PEH 135449332 Ki = 14900 nM T46814 D00YZD 54726191 IC50 > 100000 nM T46814 D01QIN 60823 IC50 = 1600 nM T46814 D01TQR 72385 Ki = 1920 nM T46814 D02EYG 10096344 IC50 > 100000 nM T46814 D02OZE 2724385 IC50 = 3235.94 nM T46814 D02RQU 54687 Ki = 3400 nM T46814 D02ZTJ 5339 Ki = 530 nM T46814 D05LYX 3488 IC50 = 1400 nM T46814 D05VIX 3463 IC50 = 11000 nM T46814 D07IQS 148192 Ki = 1300 nM T46814 D07POC 176870 IC50 = 21000 nM T46814 D07UBG 130881 Ki = 540 nM T46814 D07VLY 31703 Ki = 150000 nM T46814 D09HNR 3002190 IC50 = 3467.37 nM T46814 D09QVV 5978 Ki = 42000 nM T46814 D0AZ8C 5213 Ki = 3370 nM T46814 D0C4RB 36314 IC50 = 280 nM T46814 D0G3DL 135398735 Ki = 1100 nM T46814 D0H0ND 54454 IC50 = 4400 nM T46814 D0MY8N 5280489 Ki = 340 nM T46814 D0N6RF 65999 Ki = 1030 nM T46814 D0R0FE 2520 IC50 = 32000 nM T46814 D0R1RS 3715 Ki = 11000 nM T46814 D0W9MM 13342 Ki = 10200 nM T46814 D0Z1ZM 84029 IC50 = 3090.3 nM T46814 D0ZU9R 392622 IC50 = 700 nM T46814 D00XBC 46861584 IC50 = 398.11 nM T46814 D02AIN 122678117 IC50 = 2300 nM T46814 D0C5VQ 1548994 IC50 = 8500 nM T46814 D0CE0O 11513676 IC50 = 180 nM T46814 D0G7UX 5284373 Ki = 200 nM T46814 D0L4FS 5280961 Ki = 5000 nM T46814 D0V1WQ 24857286 IC50 = 2280 nM T46814 D0Z0HH 3503 Ki = 1780 nM T46814 D0G6ZW 636402 Ki = 1070 nM T46814 C5Q6US 2540 Ki = 400 nM T46814 CT6YF0 5100 Ki = 1430 nM T46814 C2AMP7 25096 Ki = 450 nM T46814 CYQ4S7 60822 Ki = 450 nM T46814 CXJV17 73157 Ki = 400 nM T46814 CQD56Z 73299 Ki = 2110 nM T46814 C9EQN7 73563 IC50 = 11748.98 nM T46814 C4HU6M 92095 Ki = 130 nM T46814 CNIW58 107905 Ki = 2070 nM T46814 CW90BT 441336 Ki = 1620 nM T46814 C82BDA 441371 Ki = 2410 nM T46814 CI4K8B 443953 Ki = 1670 nM T46814 CT2W6J 467315 Ki = 2050 nM T46814 C76DRY 638034 Ki = 1220 nM T46814 CAW27Q 3503223 Ki = 80 nM T46814 C8B3NE 4565183 Ki = 60 nM T46814 CT5ZR8 5149276 Ki = 620 nM T46814 CNI9X4 5281888 Ki = 4300 nM T46814 CH9WV2 5379540 Ki = 630 nM T46814 C46NFC 6426773 Ki = 260 nM T46814 CGVZ63 6708545 Ki = 380 nM T46814 C81NYO 6857763 Ki = 420 nM T46814 CAV9Q8 6857785 Ki = 1260 nM T46814 CPIV47 6857789 Ki = 2240 nM T46814 C6ROL5 6857793 Ki = 1230 nM T46814 CF5M6V 6857794 Ki = 650 nM T46814 CSH8G0 10960835 Ki = 4580 nM T46814 C7TKI8 21596329 Ki = 680 nM T46814 CM5P2W 21633776 Ki = 800 nM T46814 CYK84S 23675786 Ki = 370 nM T46814 CHJP54 23681233 Ki = 2010 nM T46814 C9P5GD 23703990 Ki = 2030 nM T46814 CPM3X9 24721251 Ki = 1820 nM T46814 C7X3WA 28330466 IC50 > 50000 nM T46814 CZ8SR1 40469657 Ki = 1940 nM T46814 CTE19R 40469671 IC50 = 1698.24 nM T46814 CKI50V 40469815 Ki = 1330 nM T46814 C70JTD 44575959 Ki = 780 nM T46814 CU49XY 52947716 Ki = 250 nM T46814 CM09JD 54676535 Ki = 590 nM T46814 C04IST 57394707 IC50 = 7943.28 nM T46814 CPE5F1 73348206 Ki = 410 nM T46814 CLAF78 73354262 Ki = 2960 nM T46814 CU3D9N 73388373 IC50 = 39810.72 nM T46814 C9R7AM 73438547 IC50 = 1400 nM T46814 CRT3Q7 76311369 Ki = 1100 nM T46814 C19WRY 76311434 Ki = 480 nM T46814 CU76LZ 76313482 Ki = 1280 nM T46814 CBLK75 76315020 Ki = 440 nM T46814 C7XM6W 76322315 IC50 = 1584.89 nM T46814 CZ8AR0 76322316 Ki = 540 nM T46814 C7W1VB 76325939 Ki = 930 nM T46814 CR6QG3 76333163 Ki = 510 nM T46814 C0T3XF 76333164 Ki = 3440 nM T46814 CE61WT 76333166 Ki = 1210 nM T46814 CQ9E0I 76336791 Ki = 830 nM T46814 C63ATV 81750201 IC50 > 50000 nM T46814 C83TUW 89825693 IC50 = 8000 nM T46814 C8LZR0 90142516 IC50 = 2800 nM T46814 CM28ET 90142544 IC50 = 4300 nM T46814 CKH7G4 90142573 IC50 = 1900 nM T46814 C0KP7T 90142592 IC50 = 2000 nM T46814 C9CVR5 90142611 IC50 = 1000 nM T46814 COVK20 90142631 IC50 = 1200 nM T46814 C7BA5F 90142659 IC50 = 1800 nM T46814 CW7I3A 90142669 IC50 = 1800 nM T46814 C4FPD3 112726150 IC50 > 50000 nM T46814 CXD39Z 118170767 IC50 = 2500 nM T46814 C9HSP6 118213818 IC50 = 3900 nM T46814 CD0TY2 118717803 IC50 = 6400 nM T46814 CHD26A 121596332 IC50 = 2000 nM T46814 C1YK2E 122678192 IC50 = 2500 nM T46814 CFB4D9 135403795 Ki = 1510 nM T46814 C7GK3H 145990715 IC50 > 100000 nM T46814 CVH0P8 155519454 IC50 = 39810.72 nM T46814 CZW45D 155525803 IC50 = 15848.93 nM T46814 CKZT21 155559364 IC50 = 1400 nM T46814 CUT84A 155568798 IC50 > 30000 nM T46814 D04LBT 14957 Ki = 2200 nM T46814 D07LUJ 64945 IC50 = 15848.93 nM T46814 D0G2JZ 1464 Ki = 18000 nM T46814 D0HD9P 444899 Ki = 330 nM T46814 D0J5RQ 234102 IC50 = 11220.18 nM T46814 D0O8ZV 5280352 Ki = 720 nM T46814 D0R4WJ 16129778 Ki = 1460 nM T46814 D0U8IF 10114 Ki = 290 nM T46814 D0UQ6U 10569 Ki = 1470 nM T31902 D01DVX 9847838 IC50 = 480 nM T31902 D0T9HG 132519 IC50 = 8.1 nM T31902 CF2T7R 2270052 IC50 > 10500 nM T31902 C1FVI6 5730271 IC50 > 10500 nM T31902 C59ZPR 5765716 IC50 = 10500 nM T31902 CQY54S 9952396 IC50 = 27 nM T31902 CY08WJ 10322755 Ki > 3000 nM T31902 CWG8Y6 11271094 IC50 = 83 nM T31902 C8C5AV 11294179 Ki > 10000 nM T31902 CK91YW 11317404 IC50 = 30 nM T31902 CN2P4G 11328571 IC50 = 58 nM T31902 C7QNX8 11363138 IC50 = 161 nM T31902 CZBF91 11476645 IC50 = 111 nM T31902 C5Z4UP 11504653 IC50 = 92 nM T31902 C5G8PM 11511807 IC50 = 18 nM T31902 C5VUM2 11517085 Ki = 734 nM T31902 C43OXZ 11519233 IC50 = 39 nM T31902 C2OA3K 11547967 IC50 = 18 nM T31902 CIWP38 11555036 IC50 = 22 nM T31902 C61BQP 11562817 IC50 = 45 nM T31902 CO9BC3 11562986 IC50 = 6.5 nM T31902 CHV2G1 11575995 Ki > 10000000 nM T31902 C3H2DG 11577137 IC50 = 44 nM T31902 CM6GO2 11577517 IC50 = 34 nM T31902 C0Q5FU 11592023 IC50 = 24 nM T31902 CSQ5M8 11598899 IC50 = 11 nM T31902 COT65V 11599397 IC50 > 1000 nM T31902 CUL5H2 11605631 IC50 = 7.1 nM T31902 CQ7G5D 11613116 IC50 = 18 nM T31902 CXKU59 11620780 IC50 = 25 nM T31902 CNY92D 11640694 Ki = 400 nM T31902 CH3V8F 11663480 IC50 = 217 nM T31902 C0WV8R 11678029 IC50 > 2000 nM T31902 CFC74O 11678245 IC50 = 14 nM T31902 CY0T4D 11685065 IC50 = 23 nM T31902 CKGR97 11692294 IC50 = 12 nM T31902 C6ORK5 11692747 IC50 > 1000 nM T31902 C3U6ZR 11697504 Ki = 29 nM T31902 C6PM1J 11713686 IC50 = 11 nM T31902 C1MJ3P 11713694 IC50 = 57 nM T31902 C4ECU2 11720597 IC50 = 286 nM T31902 C4HD9K 11751106 IC50 = 64 nM T31902 C6R1LD 15985818 IC50 = 1090 nM T31902 CD51GI 16108939 IC50 = 33 nM T31902 C5YVB0 16108940 IC50 = 137 nM T31902 CB4DU9 16108941 IC50 > 5000 nM T31902 CBW71J 16108942 IC50 = 130 nM T31902 CG6R9L 16108943 IC50 = 97 nM T31902 CN62KM 16108944 IC50 = 310 nM T31902 C7YS5Q 16108947 IC50 = 52 nM T31902 CLD2Y4 16108948 IC50 = 720 nM T31902 CJR95O 16108949 IC50 = 110 nM T31902 CRQ26L 16108950 IC50 = 330 nM T31902 CH80AG 16108951 IC50 = 23 nM T31902 CWB0G9 16108952 IC50 = 77 nM T31902 C3S2TQ 17754305 IC50 = 22 nM T31902 C5M3YW 24799779 Ki > 10000000 nM T31902 CQ2K9H 24936215 IC50 = 26 nM T31902 CA5DJ4 25138228 Ki > 10000000 nM T31902 C5S6QR 44253975 IC50 > 100000 nM T31902 CN9BZ7 44253976 IC50 = 87200 nM T31902 CY13SQ 44418977 IC50 = 480 nM T31902 C20HIJ 44446753 IC50 = 42 nM T31902 C9CS8E 44446754 IC50 = 33 nM T31902 C4Z7IQ 44446755 IC50 = 194 nM T31902 C4K5QT 44446756 IC50 = 73 nM T31902 CZEH45 44446757 IC50 = 48 nM T31902 C47SRV 44446758 IC50 = 85 nM T31902 C8CVO1 44446759 IC50 = 902 nM T31902 C8HM5N 44446763 IC50 = 28 nM T31902 CU5Z4V 44446765 IC50 = 15 nM T31902 C9USL8 44446766 IC50 = 99 nM T31902 CYO65B 44446797 IC50 = 184 nM T31902 CPI3T0 44446799 IC50 = 38 nM T31902 CGH0A2 44446805 IC50 = 14 nM T31902 CH72RW 44446806 IC50 = 1102 nM T31902 CTKX08 44446807 IC50 = 194 nM T31902 CJ1MP7 44446808 IC50 = 16 nM T31902 CJN1L7 44446821 IC50 = 68 nM T31902 C9FG5A 44446823 IC50 = 19 nM T31902 C1P0BV 44446824 IC50 = 34 nM T31902 C5AW3N 44446825 IC50 = 40 nM T31902 C17YSI 44446827 IC50 = 93 nM T31902 C3O8AX 44446835 IC50 = 19 nM T31902 CE2OM1 44446839 IC50 = 26 nM T31902 C49VJF 44446842 IC50 = 45 nM T31902 CF4DL2 44446843 IC50 = 92 nM T31902 C8OS4K 44446845 IC50 = 81 nM T31902 C6WSC7 44447346 IC50 = 102 nM T31902 C6MOB0 44447348 IC50 = 261 nM T31902 CM7JV0 44447353 IC50 = 13 nM T31902 CD8RX4 44447437 IC50 = 19 nM T31902 CLNK98 44447442 IC50 = 7.8 nM T31902 CPT42K 44580109 IC50 = 26 nM T31902 CK68GT 44580539 IC50 = 97 nM T31902 CXIY57 44580801 Ki > 10000000 nM T31902 C0OA8Y 44580802 Ki > 10000000 nM T31902 CNC4D7 44581071 Ki > 10000000 nM T31902 CDF48U 44581111 Ki > 10000000 nM T31902 C2Z4HB 44583600 IC50 = 302 nM T31902 CD4Q8C 44583601 IC50 = 19 nM T31902 CD2AQ7 44583620 IC50 = 167 nM T31902 CLZ6X5 44583621 IC50 = 77 nM T31902 C5HA4P 44583622 IC50 = 1545 nM T31902 C7PR8I 44583623 IC50 = 196 nM T31902 CDRC42 44583654 IC50 = 15 nM T31902 C5HEX6 44583655 IC50 = 165 nM T31902 CM79HD 44583656 IC50 = 21 nM T31902 C20FCM 44583672 IC50 = 915 nM T31902 CM0I4J 45101511 IC50 = 26 nM T31902 C3SQL2 45378250 IC50 = 2300 nM T31902 CO4AC6 45378252 IC50 = 240 nM T31902 C42FPG 45378253 IC50 = 190 nM T31902 CI82BN 45378254 IC50 = 2000 nM T31902 CZS39O 45487302 IC50 = 84 nM T31902 C4ZWY7 45487310 IC50 = 20 nM T31902 C9SV0H 45487311 IC50 = 30 nM T31902 C6GCM7 45487332 IC50 = 17 nM T31902 CCF05Q 45487333 IC50 = 9 nM T31902 C23NRD 45487334 IC50 = 125 nM T31902 CY09ZU 45487335 IC50 = 9.6 nM T31902 CQHJ85 45487342 IC50 = 23 nM T31902 C3ZLN1 45487343 IC50 = 12 nM T31902 CI6DW2 45487357 IC50 = 11 nM T31902 COX40Y 45487358 IC50 = 99 nM T31902 CF1T7M 45487359 IC50 = 35 nM T31902 CRXI29 45487373 IC50 = 11 nM T31902 CYL32E 45487376 IC50 = 60 nM T31902 CO5P9I 45487386 IC50 = 83 nM T31902 CS9Y8G 45487387 IC50 = 186 nM T31902 CAN4J2 45487388 IC50 = 161 nM T31902 CWLC18 45487393 IC50 = 18 nM T31902 CO9NJ2 45487398 IC50 = 14 nM T31902 CDN5Q6 45487399 IC50 = 138 nM T31902 CI4KJ5 45487400 IC50 = 20 nM T31902 C49HOI 45487401 IC50 = 58 nM T31902 CBK43U 45487402 IC50 = 78 nM T31902 C56WVI 46184724 Ki > 25000 nM T31902 CH0Z1E 46844314 Ki = 245 nM T31902 C20BTY 46856241 Ki = 166 nM T31902 C0S9WB 46919610 Ki = 602 nM T31902 C3BGW0 53233015 Ki = 1350 nM T31902 CL9SC3 54587769 Ki = 120 nM T31902 CWH7V8 57561293 IC50 = 144 nM T31902 CY1N3J 57792153 IC50 = 1211 nM T31902 C1CK0E 72714082 IC50 = 39000 nM T31902 CZFY06 72714322 IC50 = 8200 nM T31902 CDY70J 72714323 IC50 = 300 nM T31902 CD56BA 72714324 IC50 = 150 nM T31902 C5LB0U 78426619 IC50 > 100000 nM T31902 CET6N8 78426757 IC50 > 100000 nM T31902 COV8I9 86291010 IC50 = 1199 nM T31902 CAB2F5 87349434 Ki = 73 nM T31902 C1J3CK 117094707 IC50 = 40 nM T31902 CGY9V6 122181846 IC50 > 100000 nM T31902 C3GOS2 122181847 IC50 > 100000 nM T31902 CN7WC6 122181848 IC50 > 100000 nM T31902 CJ7B4Y 122181849 IC50 > 100000 nM T31902 CJNH05 122181850 IC50 > 100000 nM T31902 C2KU3W 122181851 IC50 > 100000 nM T31902 CO6N5R 122181852 IC50 > 100000 nM T31902 CN7XR8 122181988 IC50 > 100000 nM T31902 C8DHI1 122181989 IC50 > 100000 nM T31902 C9XDO5 122181990 IC50 > 100000 nM T31902 CP4M8S 122181991 IC50 > 100000 nM T31902 CT8XW5 122181992 IC50 > 100000 nM T31902 C06QZX 122181993 IC50 > 100000 nM T31902 C9G0QI 122181994 IC50 > 100000 nM T31902 C9RVB8 122181995 IC50 > 100000 nM T31902 CLCW15 122181996 IC50 > 100000 nM T31902 CT7D4F 122181997 IC50 > 100000 nM T31902 CZO32N 122181998 IC50 > 100000 nM T31902 C40DWG 122181999 IC50 > 100000 nM T31902 CT03QA 127026888 IC50 = 7000 nM T31902 CYA92R 130282633 IC50 = 950 nM T31902 CO3QE2 130282636 IC50 = 1300 nM T31902 C9CIY6 137651719 IC50 = 11700 nM T31902 CAB7Q6 137660566 IC50 > 10000 nM T31902 CF8WV2 155511139 IC50 = 5.3 nM T31902 D06EHW 11625778 IC50 = 22 nM T31902 D0A4TC 446504 IC50 = 890 nM T31902 D0VI2A 44447430 IC50 = 6.2 nM T31902 D0Y5IQ 44255320 IC50 = 10000 nM T08499 D05LYX 3488 IC50 = 12000 nM T08499 CZ0AH3 638278 IC50 = 1540 nM T08499 CR67XU 699486 IC50 = 6600 nM T08499 C4RE0S 9867803 IC50 = 210 nM T08499 CIPA47 9911728 IC50 = 260 nM T08499 CF5C8O 59847970 IC50 = 10000 nM T08499 CX5K6Q 122471062 IC50 = 2590 nM T08499 C97FVL 122499804 IC50 = 1971 nM T08499 CRE3X2 122499848 IC50 = 232 nM T08499 C7MY2H 129746657 IC50 = 42000 nM T08499 C4DS3O 134135251 IC50 = 6352 nM T08499 C64FUV 134140154 IC50 = 1828 nM T08499 CAQ4V7 134143987 IC50 = 1238 nM T08499 C8PWC6 134247765 IC50 = 5 nM T08499 C8UBG3 137515213 EC50 = 610 nM T08499 C5Q6TS 137515380 EC50 = 600 nM T08499 CNT8G1 137515383 EC50 = 220 nM T08499 CVI1H4 137515466 EC50 = 190 nM T08499 CKC32Q 137515546 EC50 = 220 nM T08499 C6Q5YE 137515571 EC50 = 220 nM T08499 CJ85ER 137515794 EC50 = 190 nM T08499 CSU98Z 137515846 EC50 = 520 nM T08499 C0M6SU 137515935 EC50 = 110 nM T08499 C4TGP3 137516041 EC50 = 240 nM T08499 CS15BK 137516054 EC50 = 860 nM T08499 C0F5XW 137516341 EC50 = 630 nM T08499 C4CA3U 145173441 IC50 = 4300 nM T08499 CX2TB3 145173449 IC50 = 3700 nM T08499 C30VAZ 145237739 IC50 = 74 nM T08499 C8I9YN 145961431 IC50 = 4800 nM T08499 CD9LY4 145961807 IC50 = 5100 nM T08499 CIG98R 145962133 IC50 = 2300000 nM T08499 CCN16I 145962393 IC50 = 3600 nM T08499 C12QYE 145963287 IC50 = 3700 nM T08499 C2EQ7Z 145964502 IC50 = 6 nM T08499 C2XDG8 145966724 IC50 = 6 nM T08499 CTP64Q 145967497 IC50 = 1220 nM T08499 CB53JT 145967694 IC50 = 15880 nM T08499 CZFI29 145970423 IC50 = 21950 nM T08499 CLD53O 145974926 IC50 = 7 nM T08499 CKBI34 145988409 IC50 = 5720 nM T08499 CRX3V8 145989045 IC50 = 39470 nM T08499 CS2G1Q 155549073 IC50 = 74000 nM T08499 D00RIX 5280443 IC50 = 10000 nM T08499 D09FGL 9910393 IC50 = 5 nM T48873 D08VRO 3822 Ki = 77 nM T48873 D0J4JM 5770 Ki = 5.26 nM T48873 D01IVE 101616 Ki = 1840 nM T48873 D0IX1I 123836 IC50 = 28.1 nM T48873 CFJ6H4 1206 IC50 = 3620 nM T48873 CFQ7R3 9345 Ki = 64 nM T48873 C3LU7J 736282 Ki = 2760 nM T48873 C81ETA 10470490 Ki = 970 nM T48873 C7DH3A 11361814 Ki = 630 nM T48873 CTH0B3 23652686 Ki = 0.1 nM T48873 CF5K0V 118691439 IC50 = 85.5 nM T48873 CW15HU 118700678 IC50 = 101 nM T48873 C5RNW2 118857804 IC50 = 39.4 nM T48873 C0GQF1 118857828 IC50 = 19.7 nM T48873 C6UHM8 118857829 Ki = 452 nM T48873 CA03SM 118857831 IC50 = 142 nM T48873 C0FCX2 118857833 Ki = 720 nM T48873 CU1Z8O 118857834 Ki = 1960 nM T48873 CX2RY8 118857835 IC50 = 125 nM T48873 C2ZD0T 118857837 Ki = 3770 nM T48873 CB54AQ 118857838 Ki = 1660 nM T48873 COT18S 145011254 IC50 = 16 nM T48873 CP9TR0 10324985 Ki > 10000 nM T48873 D0B6UU 12018178 Ki = 5160 nM T48873 D0F6CD 5202 IC50 = 1430 nM T48873 D0T6XD 10687251 Ki = 6060 nM T18784 D0L5WM 2157 IC50 = 156000 nM T18784 C2DBN5 46899607 IC50 = 1600 nM T18784 CLZ7P4 70702119 IC50 = 2232000 nM T18784 CW1GP2 70702121 IC50 = 16000 nM T18784 CI5W0K 71735843 IC50 = 200 nM T18784 C4QC5Y 145960532 IC50 = 68000 nM T18784 C8HPT2 145961258 IC50 = 102000 nM T18784 C9FGU1 145961684 IC50 = 5600 nM T18784 CF4ME6 145962269 IC50 = 86000 nM T18784 CZP8B7 145962316 IC50 = 1900 nM T18784 CJGC76 145962553 IC50 = 333000 nM T18784 CK3DZ7 145962837 IC50 = 326000 nM T18784 CVU6M3 145962898 IC50 = 76000 nM T18784 C3RB8P 145963156 IC50 = 534000 nM T18784 CK96HI 145963214 IC50 = 104000 nM T18784 C81CRJ 145963620 IC50 = 151000 nM T18784 C2WKX0 145963644 IC50 = 98000 nM T18784 D07IOY 10365 IC50 = 15000 nM T18784 D08IZY 3080614 IC50 > 250000 nM T18784 D0B2WZ 15331 IC50 = 2100 nM T12081 D01LCC 17754438 IC50 > 10000 nM T12081 D03QJL 3671 IC50 = 239 nM T12081 D09TFB 9896267 IC50 > 100 nM T12081 D0A9IY 135564558 IC50 > 10000 nM T12081 D0SM0W 44591583 IC50 = 55 nM T12081 D0T5PO 5092 IC50 = 118 nM T12081 D0Z2FB 154575 IC50 = 3.8 nM T12081 D02EMR 151170 IC50 = 610 nM T12081 D0UG4T 127928 IC50 = 4.5 nM T12081 C4B3YS 78864 IC50 = 3690 nM T12081 CFJ62Y 9799389 IC50 = 1230 nM T12081 CYXD04 9810934 IC50 = 40 nM T12081 CL70YN 9840066 IC50 = 18 nM T12081 C81LSK 9928390 IC50 = 570 nM T12081 CV6TO1 9995407 IC50 = 15.3 nM T12081 CFPR64 9999276 IC50 = 68 nM T12081 CK5C9Z 10119563 IC50 = 6.8 nM T12081 C1EVS3 10119564 IC50 = 11.4 nM T12081 C83BSD 10128917 IC50 = 1 nM T12081 CWDR26 10129145 IC50 = 17 nM T12081 CME68G 10152836 IC50 = 1.7 nM T12081 C0PVT2 10153372 IC50 = 14 nM T12081 CBT4P1 10177031 IC50 = 77 nM T12081 C3X9DK 10183196 IC50 = 22 nM T12081 CUXV40 10183769 IC50 = 3.8 nM T12081 CY9HS7 10185841 IC50 = 1.2 nM T12081 CVUZ36 10195164 IC50 = 11.9 nM T12081 C8LYH6 10196396 IC50 = 4.2 nM T12081 CSQ16M 10196596 IC50 = 9.5 nM T12081 CTV6F9 10196609 IC50 = 0.9 nM T12081 CTZ7Q8 10196916 IC50 = 6.4 nM T12081 CZG54F 10197046 IC50 = 7.5 nM T12081 C61CZK 10205978 IC50 = 68 nM T12081 CPU09I 10210579 IC50 = 14 nM T12081 CX9LV3 10232106 IC50 = 14 nM T12081 C48ENU 10289786 IC50 = 41 nM T12081 CT5FL2 10289848 IC50 = 0.05 nM T12081 CECW14 10301548 IC50 = 0.4 nM T12081 C5IF9A 10312566 IC50 = 5.9 nM T12081 C23HSK 10451184 IC50 = 190 nM T12081 C1RG7I 10545177 IC50 > 10000 nM T12081 C7G1BH 10547592 IC50 > 10000 nM T12081 CZ15HV 10571743 IC50 = 6400 nM T12081 C8RN0L 10611778 IC50 > 10000 nM T12081 CHU62M 10661230 IC50 = 890 nM T12081 CRJ79L 10664015 IC50 = 610 nM T12081 CO4AP8 10682163 IC50 > 10000 nM T12081 CF2BR1 10691724 IC50 = 4300 nM T12081 CNB35R 10805427 IC50 > 10000 nM T12081 CDL73U 10810934 IC50 = 3200 nM T12081 C0A7DI 11017241 IC50 = 135 nM T12081 C45VZC 11438405 IC50 > 16000 nM T12081 COLF16 11639342 IC50 = 6400 nM T12081 C1B4XD 11992634 IC50 > 2000 nM T12081 CPX16N 11993169 IC50 > 2000 nM T12081 C40KZA 15434926 IC50 = 700 nM T12081 C31LJY 16103072 IC50 = 2440 nM T12081 CXFT59 17757146 IC50 = 452 nM T12081 C1PZ8C 18734933 IC50 = 1378 nM T12081 C9DE6Y 20814950 IC50 = 106 nM T12081 C3M5NF 21865580 IC50 = 17 nM T12081 C4CWR6 21865595 IC50 = 70 nM T12081 C6T5NZ 21865599 IC50 = 25 nM T12081 CULE52 21865620 IC50 = 5.5 nM T12081 CINH54 21865627 IC50 = 26 nM T12081 CMHF08 22083604 IC50 = 11 nM T12081 C34FLM 22083724 IC50 = 0.7 nM T12081 CWIT18 22083784 IC50 = 2.9 nM T12081 CD48PX 23218492 IC50 = 125.9 nM T12081 C20VHK 24871823 IC50 = 6700 nM T12081 C6EQG2 24963293 IC50 > 2000 nM T12081 C5Q0IN 42647289 IC50 = 106 nM T12081 CNIE98 44143458 IC50 = 46 nM T12081 C2SLH8 44324331 IC50 = 95.2 nM T12081 CLMW27 44405467 IC50 = 5.7 nM T12081 CR05OY 44405507 IC50 = 3.3 nM T12081 C7OA9V 44405510 IC50 = 0.5 nM T12081 CFY36C 44410864 IC50 = 10.6 nM T12081 CT1JW4 44410870 IC50 = 1.7 nM T12081 C3EI4T 44410882 IC50 = 490 nM T12081 C7NKA2 44410914 IC50 = 97 nM T12081 C3P2IN 46933992 IC50 = 151 nM T12081 CB2HS9 46933993 IC50 = 32.2 nM T12081 CZ7C3F 46933994 IC50 = 36.2 nM T12081 C0EH7V 49865602 IC50 = 1977 nM T12081 C89UPD 49865603 IC50 = 28300 nM T12081 CV81PG 49865604 IC50 = 1235 nM T12081 C43XGJ 49865605 IC50 = 1115 nM T12081 CIT05Z 49865642 IC50 = 1341 nM T12081 C5OI1V 49865643 IC50 = 103 nM T12081 C19JZB 49866243 IC50 = 69.5 nM T12081 CU5B8G 49866268 IC50 = 31.2 nM T12081 CSYL46 49866269 IC50 = 469 nM T12081 CI3F7K 49866270 IC50 = 102.1 nM T12081 C7V8DY 49866271 IC50 = 218 nM T12081 CCJ7I1 49866272 IC50 = 414 nM T12081 CD52CA 57391118 IC50 > 2000 nM T12081 CWX3N7 59320301 IC50 = 1970 nM T12081 C0EP5I 59341847 IC50 = 2080 nM T12081 CHQ28A 59341978 IC50 = 3260 nM T12081 CJ62MK 71451776 IC50 = 206 nM T12081 C2UK6B 71451779 IC50 = 505 nM T12081 CJ3Z7K 71460703 IC50 = 10 nM T12081 CBM61I 73293715 IC50 = 2910 nM T12081 CW2HR1 130366728 IC50 = 31.4 nM T12081 C2ALN7 130366739 IC50 = 104 nM T12081 CQJN83 130366758 IC50 = 653 nM T12081 CDAF16 130380472 IC50 = 389 nM T12081 C18KLO 130380505 IC50 = 48.2 nM T12081 C5XCO1 130380512 IC50 = 108 nM T12081 CT2E8Q 130380575 IC50 = 160 nM T12081 C2P1IU 134129996 IC50 = 400 nM T12081 CLE03O 134130328 IC50 = 294 nM T12081 CSN6J0 134130563 IC50 = 269 nM T12081 C0A1CZ 134131162 IC50 = 501 nM T12081 C3R8SE 135457869 IC50 > 10000 nM T12081 CTX54Z 135896326 IC50 > 10000 nM T12081 C12UMG 136059728 IC50 > 1000 nM T12081 CLN2U7 137652270 IC50 > 10000 nM T12081 C1S7HV 142592633 IC50 = 156 nM T12081 CN3OC2 142592634 IC50 = 57 nM T12081 CY64NR 142592636 IC50 = 39 nM T12081 C83XNL 142592649 IC50 = 77 nM T12081 C7XZB1 142592652 IC50 = 326 nM T12081 C9SH7Y 145949856 IC50 > 17000 nM T12081 D01RUN 448055 IC50 = 3690 nM T12081 D02NKD 10711281 IC50 = 2000 nM T12081 D06NIT 135564899 IC50 > 1000 nM T12081 D0JD4C 9853498 IC50 = 9.1 nM T12081 D0P2TS 9818682 IC50 = 2400 nM T12081 D0V4WB 149790 IC50 > 16000 nM T12081 D0W7WV 11039077 IC50 = 1 nM T53159 D02TUL 118115473 IC50 > 50000 nM T53159 D0E3TC 44259 IC50 = 1280 nM T53159 D03BNU 59604787 IC50 > 10000 nM T53159 CK2J3G 9863776 IC50 = 300 nM T53159 C0APW4 11422034 IC50 > 10000 nM T53159 C1ZPM5 11630874 IC50 > 10000 nM T53159 CJ9KN7 11683817 IC50 > 10000 nM T53159 CU0E8O 11690457 Ki > 2000 nM T53159 CB0AP2 11705863 Ki > 10000 nM T53159 C9TU1O 16046126 IC50 > 1000 nM T53159 C5Z3LI 44591740 IC50 = 860 nM T53159 C1MR8Q 60097495 IC50 > 10000 nM T53159 CZ4BX1 72547959 IC50 > 5000 nM T53159 CJQ5N6 91936970 IC50 > 5000 nM T53159 C3Z4AT 137321159 IC50 > 10000 nM T53159 C28QUP 137652864 IC50 = 188.6 nM T53159 CE31VG 145979714 IC50 > 10000 nM T53159 C9BX4U 145988956 IC50 > 10000 nM T53159 C2MD1Q 155513187 IC50 > 10000 nM T63220 D0AF6O 71731823 IC50 = 17 nM T63220 D0E6XR 3062316 Ki < 10 nM T63220 D0OB0F 5328940 IC50 = 2.7 nM T63220 D03HUX 49792852 IC50 > 10000 nM T63220 D0E3TC 44259 IC50 = 34.8 nM T63220 D0O0LS 25141092 IC50 = 70 nM T63220 D03BNU 59604787 IC50 > 10000 nM T63220 D0PX1D 57961044 IC50 = 58 nM T63220 D0SZ3I 44468332 IC50 = 84 nM T63220 D0T9JA 44538590 IC50 = 170 nM T63220 CM9GA6 290208 Ki = 1000 nM T63220 CUJR40 10062694 IC50 = 18 nM T63220 CE36DN 11156201 IC50 = 35 nM T63220 CJ5W9L 11181283 IC50 = 20 nM T63220 C3TOH4 11191242 IC50 = 21 nM T63220 C0YH2X 11478363 IC50 = 25 nM T63220 C8RQD7 11501591 IC50 = 24 nM T63220 C87ARG 11519208 IC50 = 20 nM T63220 CHW13Q 11519350 IC50 = 38 nM T63220 CTG83F 11539329 Ki > 9500 nM T63220 CX06WK 11545532 Ki > 10000 nM T63220 C32PUD 11553058 IC50 = 420 nM T63220 CW43OA 11554885 IC50 = 148 nM T63220 CJ59WD 11562553 IC50 = 332 nM T63220 C4O9VX 11576813 Ki = 0.3 nM T63220 CMIL86 11590363 Ki > 9500 nM T63220 C45BMY 11603130 Ki = 70 nM T63220 CU6T2L 11613133 IC50 = 84 nM T63220 CUQ4I5 11620266 IC50 = 91 nM T63220 CG1JN5 11620467 IC50 = 170 nM T63220 C9ZD2E 11626406 IC50 = 78 nM T63220 CX72ET 11626681 IC50 = 650 nM T63220 CPB48V 11626947 IC50 = 97 nM T63220 C7CV8O 11634876 IC50 = 85 nM T63220 C1TZY3 11635079 IC50 = 150 nM T63220 C9T6SC 11640926 Ki > 9500 nM T63220 CA80WI 11648745 IC50 = 17 nM T63220 C82TKN 11656437 IC50 = 13 nM T63220 C3L2HT 11656560 IC50 = 930 nM T63220 CX7C1T 11656606 IC50 = 120 nM T63220 C60ASI 11663230 Ki = 0.2 nM T63220 C8RMT2 11663885 IC50 = 180 nM T63220 C1LV6H 11677453 IC50 = 16 nM T63220 CA4Q5F 11678465 IC50 = 586 nM T63220 CP3U0W 11684933 IC50 = 98 nM T63220 CYO6X9 11684994 Ki = 0.3 nM T63220 CI3EO4 11692100 IC50 = 180 nM T63220 CZV0O2 12003241 IC50 = 9 nM T63220 CLR3S1 15965424 Ki = 2 nM T63220 CFPW41 16007116 Ki > 9500 nM T63220 C65FUM 16048823 Ki = 30 nM T63220 C68YHJ 16048825 Ki = 40 nM T63220 C2UZJ0 16048826 Ki = 100 nM T63220 C9NSM1 16048974 Ki = 50 nM T63220 CZ61VI 16048979 Ki = 3 nM T63220 CVS24I 16049186 Ki > 4000 nM T63220 C17XEN 16049187 Ki = 400 nM T63220 C6F7QU 16049188 Ki > 2500 nM T63220 CASB59 16049257 Ki = 26 nM T63220 C67ZPN 16049258 Ki = 18 nM T63220 CAY9H0 16049260 Ki = 2 nM T63220 C5VPH9 16129448 IC50 = 558 nM T63220 C28TDB 17756743 IC50 = 181 nM T63220 CSO82D 25154877 Ki = 3 nM T63220 CW1S4G 25154878 Ki = 10 nM T63220 CRO8T9 25263033 Ki = 3 nM T63220 CN8WB9 44189332 IC50 = 149 nM T63220 CL05KJ 44438314 IC50 = 523 nM T63220 C3XQK1 44438318 Ki = 5 nM T63220 CSB51N 44438320 IC50 = 7 nM T63220 CO7PI2 44438839 IC50 = 190 nM T63220 CI8YZ1 44538074 IC50 = 1900 nM T63220 C1O4CY 44538587 IC50 = 130 nM T63220 C9N1BU 44539192 IC50 = 35 nM T63220 CXMQ28 44539284 IC50 = 87 nM T63220 CS75OB 44539383 IC50 = 570 nM T63220 CGKD81 44539384 IC50 = 380 nM T63220 CKIW24 44539387 IC50 = 90 nM T63220 C3VRO9 44557921 IC50 > 10000 nM T63220 CY76QW 44562670 Ki = 30 nM T63220 C3XTA7 44562721 Ki = 20 nM T63220 C9K2FL 44562722 Ki = 12 nM T63220 CB8S7M 44562723 Ki = 10 nM T63220 C25BGD 44562724 Ki = 30 nM T63220 C0QTD8 44562725 Ki = 80 nM T63220 C8PW4X 44562974 IC50 = 2 nM T63220 CW0M8G 44562975 Ki = 7 nM T63220 CU7C3Z 44563015 Ki = 10 nM T63220 C70OMS 44563016 Ki = 2 nM T63220 CP1C6L 44563017 Ki = 30 nM T63220 CI5SO9 44563018 Ki = 10 nM T63220 CJ8X6O 44563019 Ki = 30 nM T63220 C9BH6Q 44563020 Ki = 70 nM T63220 CD7O6M 44563040 Ki = 5 nM T63220 C3F0IA 44563041 Ki = 5 nM T63220 CU3RF1 45139989 IC50 > 10000 nM T63220 CQGZ06 45139991 IC50 > 10000 nM T63220 C7ON5A 46233287 IC50 > 10000 nM T63220 CWM9H3 46900076 IC50 = 37 nM T63220 CF91RS 49843531 IC50 > 10000 nM T63220 C2Y6QS 50938552 IC50 > 10000 nM T63220 C9NYP4 51036677 IC50 > 10000 nM T63220 C4WRY3 51037112 IC50 > 10000 nM T63220 CRI28Z 51037948 IC50 > 10000 nM T63220 COZ6H9 57960797 IC50 = 240 nM T63220 CE7X5Z 57960805 IC50 = 5460 nM T63220 C4R1VN 57960806 IC50 = 470 nM T63220 C65PAR 57960830 IC50 = 88 nM T63220 CT4U2Q 57960837 IC50 = 220 nM T63220 CDB27Q 57960863 IC50 = 240 nM T63220 CH3IR5 57960867 IC50 = 4090 nM T63220 CC9VW5 57960887 IC50 = 330 nM T63220 C57GMX 57960888 IC50 = 110 nM T63220 C3MLW4 57960890 IC50 = 48 nM T63220 C6FCA7 57960901 IC50 = 160 nM T63220 CZ65CH 57960904 IC50 > 10000 nM T63220 C4J5KC 57960906 IC50 = 1060 nM T63220 CA8F5H 57960910 IC50 = 1690 nM T63220 CLR7V6 57960920 IC50 = 3190 nM T63220 CZTM16 57960930 IC50 = 740 nM T63220 CD6Q0J 57960960 IC50 = 88 nM T63220 C85NPU 57960964 IC50 = 29 nM T63220 CY0I4P 57960972 IC50 = 100 nM T63220 CO1D0J 57960986 IC50 = 370 nM T63220 C93NVL 57960992 IC50 = 30 nM T63220 C41OVB 57961010 IC50 = 75 nM T63220 C61FIH 57961014 IC50 = 1870 nM T63220 CCAZ13 57961015 IC50 > 10000 nM T63220 C30AJR 57961033 IC50 = 900 nM T63220 C15VRC 57961037 IC50 = 3350 nM T63220 CX6PA8 57961047 IC50 = 6280 nM T63220 CCW3Z9 58603248 Ki = 6 nM T63220 CW5R1T 58603258 Ki = 4 nM T63220 C61QTX 58603262 Ki = 10 nM T63220 COV07M 58603296 Ki = 8 nM T63220 CH7QC2 58603322 Ki = 13 nM T63220 CKN1V2 58603337 Ki = 40 nM T63220 C16FRW 58603341 Ki = 20 nM T63220 C3WT0Q 58603342 Ki = 2 nM T63220 C83YSL 58603344 Ki = 6 nM T63220 C9Q4OG 58603347 Ki = 30 nM T63220 C9OS6G 58603350 Ki = 3 nM T63220 CR8T3P 59711970 IC50 = 60 nM T63220 C37NKO 67129970 IC50 = 3460 nM T63220 CK80LJ 67130050 IC50 = 1320 nM T63220 CV63UL 67240318 IC50 > 10000 nM T63220 C0LHY7 68458136 Ki = 8 nM T63220 C7GRV2 68755406 IC50 = 4020 nM T63220 C5XLE3 70682725 Ki = 6 nM T63220 CJH92U 70682726 Ki = 2 nM T63220 CC31EK 70684805 Ki = 7 nM T63220 C4Z6EW 70684806 Ki = 2 nM T63220 C9XR8I 70684807 Ki = 4 nM T63220 CXN79V 70684808 Ki = 20 nM T63220 CBZ7P6 70684809 Ki = 1980 nM T63220 CCTV49 70684823 Ki = 4 nM T63220 CP4W6Y 70684824 Ki = 50 nM T63220 CQ58YR 70686968 Ki = 40 nM T63220 CYK4A1 70686985 Ki = 4 nM T63220 CFS5V7 70689045 Ki = 69 nM T63220 C40XZG 70689046 Ki = 7300 nM T63220 CWVN64 70691142 Ki = 5 nM T63220 C3RGT8 70691155 Ki = 20 nM T63220 CXQJ05 70693256 Ki = 6 nM T63220 C3QRE1 70693257 Ki = 4 nM T63220 CNJ71U 70693258 Ki = 6 nM T63220 CL05RF 70693268 Ki = 50 nM T63220 C0Q1RX 70693269 Ki = 1800 nM T63220 C5QNW0 70695344 Ki = 6 nM T63220 CM18HU 70695345 Ki = 4 nM T63220 C1PAO5 70695346 Ki = 10 nM T63220 CE4F8O 70695358 Ki = 13 nM T63220 CP9G4T 70697354 Ki = 6 nM T63220 CH9TK3 70697355 Ki = 10 nM T63220 CCN01X 71547862 IC50 > 10000 nM T63220 C82PYL 71553074 IC50 > 10000 nM T63220 CQM7W5 71553143 IC50 = 280 nM T63220 CZM1K4 71765510 IC50 = 11 nM T63220 C0DL3F 72698602 IC50 = 14.27 nM T63220 CFB75T 90479825 IC50 = 56 nM T63220 CY0UC4 90645194 IC50 > 10000 nM T63220 CR0N6B 117857501 IC50 = 53.3 nM T63220 C3H4UB 117857550 IC50 = 85 nM T63220 C76YVZ 117857773 IC50 = 48.3 nM T63220 C47FUO 117857779 IC50 = 299 nM T63220 C9Y5DG 117857786 IC50 = 164 nM T63220 CWUQ12 117858124 IC50 = 33.2 nM T63220 C2PT1G 117858190 IC50 = 99 nM T63220 CWF6J7 117858229 IC50 = 231 nM T63220 C3HPG4 117858443 IC50 = 169 nM T63220 C8BK7O 117859438 IC50 = 82 nM T63220 C6Q8DS 117859439 IC50 = 54.4 nM T63220 C10QRJ 117859462 IC50 = 48 nM T63220 CE50FX 117859566 IC50 = 94.7 nM T63220 C02IWF 117859613 IC50 = 54.4 nM T63220 C4RU6F 117859653 IC50 = 47.7 nM T63220 CQH9V8 117864043 IC50 = 106 nM T63220 CG87BL 117864051 IC50 = 67.5 nM T63220 CO1P9Q 117864057 IC50 = 81.3 nM T63220 CRN6G4 117864062 IC50 = 34.2 nM T63220 CY7BI2 118706214 IC50 > 10000 nM T63220 C4TX7F 118737443 IC50 = 28.4 nM T63220 CM3WO6 134304664 IC50 = 28 nM T63220 CR6L0B 134304723 IC50 = 20 nM T63220 CJI0G1 135520135 IC50 > 10000 nM T63220 CHA4N2 136013680 IC50 > 10 nM T63220 CH64ID 136175114 IC50 > 10000 nM T63220 C1YUD0 136219394 IC50 > 10 nM T63220 CIU8W3 136254389 IC50 > 10 nM T63220 CSGM03 137210056 IC50 > 10000 nM T63220 CXC69T 137321158 IC50 = 995 nM T63220 CXP53D 137348835 IC50 = 8 nM T63220 CI1E8V 137634241 IC50 = 1330 nM T63220 C49KUQ 145964145 IC50 = 10 nM T63220 CE5S1W 145964374 IC50 = 53 nM T63220 CPVG78 145964598 IC50 = 28 nM T63220 C9MX1N 145964844 IC50 = 20 nM T63220 CP83FM 145964889 IC50 = 36 nM T63220 CL3H4Z 145965408 IC50 = 21 nM T63220 CSK06W 145966254 IC50 = 21 nM T63220 CWK7C2 145966484 IC50 = 11 nM T63220 C6RXU9 145967106 IC50 = 94 nM T63220 CK0CV9 145970783 IC50 = 26 nM T63220 C0Y2WF 145972806 IC50 = 15 nM T63220 CAGL67 145972836 IC50 = 25 nM T63220 C4J5YX 145976700 IC50 = 25 nM T63220 CF6NW2 145976762 IC50 = 23 nM T63220 C5RX9K 145977177 IC50 = 26 nM T63220 CJE14S 145977878 IC50 = 40 nM T63220 CJ07WY 145978202 IC50 = 13 nM T63220 C75UKW 145978330 IC50 = 40 nM T63220 CN58FM 145978369 IC50 = 6 nM T63220 C2MD1Q 155513187 IC50 > 10000 nM T63220 C78MZC 155536330 IC50 = 13 nM T63220 D00HVA 11624601 Ki > 9500 nM T63220 D09HVH 135566652 IC50 > 10 nM T63220 D09PTP 57325421 IC50 = 41 nM T63220 D0D5KZ 11540659 IC50 = 1 nM T63220 D0K5UF 72710568 IC50 = 15 nM T63220 D0Q3NG 11715520 Ki > 9500 nM T63220 D0S7IE 11658882 Ki > 9500 nM T83369 D03QJN 9895762 Ki = 2200 nM T83369 D0D5RH 11641515 IC50 = 4500 nM T83369 D0K1PR 1747 Ki = 950 nM T83369 CY5B9C 1504 Ki = 99 nM T83369 CZP0Y1 204101 Ki = 9000 nM T83369 C0KI2N 5287439 Ki = 13 nM T83369 C7SYK9 6102731 IC50 = 44 nM T83369 CX34ZD 9549214 Ki > 1800 nM T83369 C2AXV0 9809479 Ki > 41000 nM T83369 CC0D5H 9915041 Ki > 12000 nM T83369 C8F5CW 9937921 Ki = 2200 nM T83369 C8LR4T 9938917 Ki > 15000 nM T83369 C31QAL 10143532 Ki > 12000 nM T83369 CFIH78 10185526 IC50 = 51 nM T83369 CQ9ZO1 10275412 Ki > 15000 nM T83369 CJ28HS 10325481 Ki = 59 nM T83369 CEI65Z 10483775 Ki > 20000 nM T83369 CRDU42 11271947 Ki > 33000 nM T83369 CVI82D 11479420 Ki = 3500 nM T83369 CJP9O1 11684611 Ki > 34900 nM T83369 CNZ04Q 11740591 Ki > 3000 nM T83369 CX5S1Z 15511974 Ki = 6700 nM T83369 C7VH6K 15950345 Ki > 12000 nM T83369 CA8Y1K 16046152 Ki > 41000 nM T83369 CNBJ60 16046153 Ki > 41000 nM T83369 C63ILO 18549509 Ki = 72 nM T83369 CERC13 19007351 Ki = 8000 nM T83369 CZ6KH9 20760195 Ki > 15000 nM T83369 CEL6C2 23644671 Ki = 82 nM T83369 CM01LP 23646188 Ki = 11 nM T83369 CA3U0I 23646189 Ki = 7.9 nM T83369 CIR65F 23646190 Ki = 8 nM T83369 CDK0P2 23646191 Ki = 7.9 nM T83369 CJ4U2X 23646192 Ki = 13 nM T83369 CMYI38 23646193 Ki = 4.2 nM T83369 CZ1KO7 23646194 Ki = 5.1 nM T83369 CPF54M 23646195 Ki = 6.4 nM T83369 CP84AB 23646196 Ki = 10 nM T83369 C2WK4G 23646197 Ki = 11 nM T83369 CC1FV9 23646198 Ki = 11 nM T83369 CG82YE 23646199 Ki = 26 nM T83369 C5KWB9 23646200 Ki = 1700 nM T83369 CY8SQ7 23646201 Ki = 190 nM T83369 CCMZ94 23646202 Ki = 120 nM T83369 C08AOH 23646204 Ki = 20 nM T83369 C82COD 23646205 Ki = 11 nM T83369 CS5AL3 23646206 Ki = 5.5 nM T83369 C0EO5K 23646207 Ki = 15 nM T83369 CN1Q7D 23646208 Ki = 660 nM T83369 CP24HW 23646209 Ki = 63 nM T83369 C6UM7B 23646210 Ki = 19 nM T83369 C7NKV6 23646211 Ki = 820 nM T83369 CGB18F 23646212 Ki = 480 nM T83369 C5J3OT 23646213 Ki = 750 nM T83369 C3JF1O 23646214 Ki = 160 nM T83369 C75SDV 23646215 Ki = 3800 nM T83369 C8G0NU 23646216 Ki = 240 nM T83369 C84HGM 23646217 Ki = 98 nM T83369 CATE50 23646218 Ki = 75 nM T83369 CC52RE 23646219 Ki = 1200 nM T83369 C7CZ2J 23646220 Ki = 270 nM T83369 CLDZ20 23646221 Ki = 130 nM T83369 CM7X3R 23646222 Ki = 300 nM T83369 CG3ZB2 23646223 Ki = 360 nM T83369 CQS7X6 23646224 Ki = 130 nM T83369 CHAD98 23646225 Ki = 250 nM T83369 C8XZ3J 23646226 Ki = 310 nM T83369 CP9A1B 23646227 Ki = 930 nM T83369 CJS63R 23646228 Ki = 1900 nM T83369 CJN96Y 23646229 Ki = 270 nM T83369 C01VKP 23646230 Ki = 660 nM T83369 CL14AX 23646231 Ki = 98 nM T83369 C96UDO 23646233 Ki = 63 nM T83369 C6RM8B 23646234 Ki = 74 nM T83369 C2U0RB 23646236 Ki = 75 nM T83369 CPMW70 23646237 Ki = 230 nM T83369 CS5CV9 23646239 Ki = 220 nM T83369 CV1HY5 23646241 Ki = 4900 nM T83369 C6BG3M 23646243 Ki = 1250 nM T83369 CU2V7C 23646245 Ki = 390 nM T83369 C93IYD 23646247 Ki = 930 nM T83369 C5LQ0H 23646249 Ki = 250 nM T83369 CS68GZ 23646251 Ki = 780 nM T83369 C7FEL6 23646252 Ki = 1730 nM T83369 C3ZAY1 23646254 Ki = 960 nM T83369 C6EF4Y 23646256 Ki = 580 nM T83369 CKM7Y4 23646258 Ki = 130 nM T83369 C0UMW5 23646268 Ki = 480 nM T83369 C2RV5T 23646269 Ki = 14220 nM T83369 CRX19I 23646295 Ki > 12000 nM T83369 CCRD27 23646312 Ki = 37000 nM T83369 C1WE6B 23646315 Ki > 41000 nM T83369 CJSO87 24849206 Ki > 33000 nM T83369 CN0ZW3 24999867 Ki > 1000 nM T83369 CEM32W 25001205 Ki > 1000 nM T83369 C2H4PJ 25166809 Ki > 73000 nM T83369 CESM50 44392171 Ki = 1190 nM T83369 CRYN03 44392172 Ki = 310 nM T83369 C9FUI3 44392182 Ki > 120 nM T83369 CT1AO2 44392186 Ki = 500 nM T83369 CG8V4B 44392189 Ki = 8530 nM T83369 CVK58T 44392197 Ki = 430 nM T83369 C4CU6F 44392199 Ki = 280 nM T83369 C1K6IY 44392201 Ki > 32000 nM T83369 CKO0E4 44392205 Ki = 240 nM T83369 CAE80C 44392206 Ki = 280 nM T83369 CJC84M 44392224 Ki = 41300 nM T83369 CP1CF2 44392233 Ki = 3500 nM T83369 CHQG45 44392249 Ki = 340 nM T83369 C45EDM 44392250 Ki = 140 nM T83369 CUFO09 44395404 Ki = 44 nM T83369 C3BX5Y 44412781 Ki > 150000 nM T83369 C4A8IF 44422910 Ki = 1240 nM T83369 CVZW52 44537923 IC50 = 17000 nM T83369 C7K6JN 44587263 Ki > 100000 nM T83369 CDBV80 44587292 Ki > 100000 nM T83369 C4LQW3 44629430 Ki = 5900 nM T83369 CUK2I7 45103480 Ki = 140 nM T83369 CP6SB1 45103481 Ki = 130 nM T83369 CM16YW 45103482 Ki = 140 nM T83369 CKN2F4 45103582 Ki = 420 nM T83369 C80DXA 45103583 Ki = 290 nM T83369 CG51EA 45103584 Ki = 340 nM T83369 C46JPW 45103585 Ki = 100 nM T83369 C8XBZ6 45103586 Ki = 50 nM T83369 CXS6K8 45103587 Ki = 4 nM T83369 CPR1O7 45103680 Ki = 3 nM T83369 CJU8M5 45103681 Ki = 8 nM T83369 C9L1ZS 46233075 Ki = 9 nM T83369 CD62VO 46233076 Ki = 5 nM T83369 C5PI6E 46233077 Ki = 11 nM T83369 C9BLH7 46233114 Ki = 5 nM T83369 C42DOH 46233115 Ki = 3 nM T83369 CA7S2F 46233116 Ki = 15.5 nM T83369 CQ4UF5 46233117 Ki = 4.4 nM T83369 CEU41B 46233150 Ki = 8.1 nM T83369 CXV4P6 46233151 Ki = 270 nM T83369 C7WDV1 46233152 Ki = 11900 nM T83369 CFA7H0 46233153 Ki = 800 nM T83369 CH01MJ 46233194 Ki = 3800 nM T83369 C97GVT 46233259 Ki = 24200 nM T83369 CKC4V9 46233260 Ki = 23000 nM T83369 CR5VN4 46233261 Ki = 680 nM T83369 CHF74W 46233262 Ki = 700 nM T83369 C9AC2K 46233263 Ki = 7200 nM T83369 C8ONP6 46233306 Ki = 900 nM T83369 CG6QI5 46233307 Ki = 450 nM T83369 CD5K9T 46233308 Ki = 26900 nM T83369 CL0W5E 46233309 Ki = 450 nM T83369 C8AQZ5 46233310 Ki = 250 nM T83369 C7XT0F 46233339 Ki = 900 nM T83369 C7LE2Q 46233340 Ki = 11300 nM T83369 CJ3P5N 46233341 Ki = 450 nM T83369 CBC4Y5 46233342 Ki = 75 nM T83369 CUPC52 46233343 Ki = 31 nM T83369 CHF45Z 46233364 Ki = 5150 nM T83369 C2SR3C 46233365 Ki = 21600 nM T83369 CUZW20 46233366 Ki = 1050 nM T83369 CTMN13 46233367 Ki = 350 nM T83369 CA36GE 46233368 Ki = 11300 nM T83369 C23KIW 46233369 Ki = 1980 nM T83369 CLHX82 46233406 Ki = 500 nM T83369 C8Y2GA 46233407 Ki = 8400 nM T83369 C8T5CW 46233408 Ki = 1000 nM T83369 CQ01MF 46233409 Ki = 170 nM T83369 CY92TG 46233410 Ki = 390 nM T83369 CZ7CQ8 46233411 Ki = 40 nM T83369 CPBS35 46233412 Ki = 21 nM T83369 C12SEZ 46233413 Ki = 20 nM T83369 C7VKZ8 46233414 Ki = 28 nM T83369 CCI75A 46233462 Ki = 36 nM T83369 CYG6A2 46233463 Ki = 3 nM T83369 CT5MH6 46233491 Ki = 370 nM T83369 CY5C1O 46233492 Ki = 160 nM T83369 C5H2EF 46233511 Ki = 29 nM T83369 CZ46CU 46233512 Ki = 270 nM T83369 CI8NV4 46233513 Ki = 97 nM T83369 C84HTG 46233514 Ki = 28 nM T83369 CA4Z5X 46233537 Ki = 10 nM T83369 C5SK7C 46233538 Ki = 61 nM T83369 C0Y8IT 46233539 Ki = 5 nM T83369 C16IMD 46233540 Ki = 25 nM T83369 CW3S0U 46233565 Ki = 8 nM T83369 C03TRU 46233566 Ki = 8 nM T83369 C8RCY2 46233567 Ki = 5 nM T83369 CHO28I 46233568 Ki = 3 nM T83369 CRDC20 46233603 Ki = 35 nM T83369 CWVY84 46233604 Ki = 4 nM T83369 C7ZP4M 46233605 Ki = 10 nM T83369 CT84CW 46233649 Ki = 3 nM T83369 CF8Z3Q 46233651 Ki = 8 nM T83369 CX28UI 46233688 Ki = 7 nM T83369 C9P0FC 46233689 Ki = 7 nM T83369 CWO0V7 46233690 Ki = 12 nM T83369 C7ET8Q 46233691 Ki = 10 nM T83369 CB2F7T 46978227 Ki = 9000 nM T83369 CLOY62 49864459 Ki > 33000 nM T83369 CR8JK9 49864483 Ki > 33000 nM T83369 CA6GQ5 53341037 Ki > 27100 nM T83369 C0CZ7B 54726725 Ki = 120000 nM T83369 CTE30K 57842560 Ki > 35000 nM T83369 C0C6UB 57842624 Ki > 35000 nM T83369 C7XY5A 57842673 Ki > 35000 nM T83369 C41NSR 57842812 Ki = 34000 nM T83369 CWF0C3 57842850 Ki > 35000 nM T83369 C73CPB 57842913 Ki = 16000 nM T83369 C60HCV 57976401 Ki > 27100 nM T83369 CM8UJ7 57976444 Ki > 35000 nM T83369 CQ71KE 57976446 Ki > 60000 nM T83369 CSC0L5 59020200 Ki > 15000 nM T83369 C91APY 59095797 IC50 = 66 nM T83369 C69SED 59095888 IC50 = 180 nM T83369 CYB84G 59095944 IC50 = 1800 nM T83369 CO38AC 59402011 Ki > 73000 nM T83369 CE5A7B 60162406 Ki > 100000 nM T83369 CWCA65 66573845 IC50 > 1000000 nM T83369 CWOD93 66744646 Ki > 27100 nM T83369 CKWQ82 67155200 Ki = 34200 nM T83369 CA49UK 69520512 Ki > 29000 nM T83369 CTO5I6 70253788 Ki = 39300 nM T83369 C9EL3C 71260387 Ki > 27100 nM T83369 CJPF90 71548883 Ki > 27000 nM T83369 C30ZKJ 71561420 Ki > 5000 nM T83369 C83ZNH 71562308 IC50 = 1141 ug.mL-1 T83369 C62ZTJ 71660643 IC50 = 20000 nM T83369 CVM7Y6 71748093 Ki = 15000 nM T83369 C6CB0G 71748095 Ki = 15000 nM T83369 C3DWZ2 72163854 IC50 = 6700 nM T83369 CRBH34 72164200 IC50 = 13 nM T83369 CWNZ45 72164201 IC50 = 67 nM T83369 CLI36U 72551247 Ki = 1600 nM T83369 CAT95V 76685067 IC50 > 100000 nM T83369 CMD5V7 86583041 Ki > 34860 nM T83369 CO6U9I 88582319 Ki > 73700 nM T83369 CUC01L 91799239 Ki = 3.6 nM T83369 CE28SQ 91972030 IC50 = 98 nM T83369 CYH43T 118456915 IC50 = 45 nM T83369 CM39QL 118456920 IC50 = 15 nM T83369 C1C3HV 118456930 IC50 = 32 nM T83369 CKST03 118456931 IC50 = 13 nM T83369 C4CJM6 118456935 IC50 = 18 nM T83369 C6EJB5 118456946 IC50 = 32 nM T83369 C6ZS9A 118456950 IC50 = 33 nM T83369 CQ43TO 118456975 IC50 = 47 nM T83369 CL4K5X 118456998 IC50 = 172 nM T83369 CCR4Y5 118457019 IC50 = 13 nM T83369 C26CAL 118457021 IC50 = 26 nM T83369 COY1V8 118457032 IC50 = 62 nM T83369 CWY2B9 118457044 IC50 = 36 nM T83369 CS05DP 118457052 IC50 = 89 nM T83369 CKS29X 118713018 IC50 > 100000 nM T83369 CRF62H 118713026 IC50 > 100000 nM T83369 CAS3L5 118713029 IC50 > 100000 nM T83369 CRV5Y1 118721008 Ki > 34900 nM T83369 CNPK35 118736105 Ki = 114000 nM T83369 CL1B0F 118736106 Ki = 8520 nM T83369 CF2B3P 118736107 Ki = 7760 nM T83369 C0GVT6 118736108 Ki = 32200 nM T83369 C9Y1TE 118736109 Ki = 86600 nM T83369 C76FAD 118736110 Ki > 145000 nM T83369 CX4R9M 118736111 Ki = 54200 nM T83369 CVW51N 118736112 Ki = 131000 nM T83369 CJTB51 118736113 Ki > 145000 nM T83369 C6FYE4 118736114 Ki > 145000 nM T83369 C79CNJ 118736115 Ki > 145000 nM T83369 CMH15Y 118736116 Ki = 2040 nM T83369 C2CKP6 118736117 Ki = 18800 nM T83369 CP17DN 118736118 Ki > 145000 nM T83369 CZMQ94 118736119 Ki = 260 nM T83369 CDHA74 118736120 Ki = 2120 nM T83369 CC72ML 118736121 Ki = 130000 nM T83369 CW3X2A 118736122 Ki > 145000 nM T83369 CGA34B 118736123 Ki = 5580 nM T83369 CHG9B7 118736124 Ki = 462 nM T83369 CPH87E 118736125 Ki = 2000 nM T83369 C5DEU9 118736126 Ki = 18300 nM T83369 CU7N0O 118736127 Ki = 20600 nM T83369 CA1YT2 118736128 Ki = 6340 nM T83369 C32KLW 118736129 Ki = 90 nM T83369 C0J8QU 118736130 Ki = 156 nM T83369 CKCW81 118736131 Ki = 937 nM T83369 CFWI73 118736132 Ki = 30300 nM T83369 CDAR13 118736133 Ki = 595 nM T83369 C13SZX 118736134 Ki = 4400 nM T83369 CLO4M2 118736135 Ki = 55400 nM T83369 C4X7SG 118736136 Ki = 35000 nM T83369 C8H5SO 118736137 Ki = 340 nM T83369 CPN2Q3 118736138 Ki = 15.7 nM T83369 CI89KX 118736139 Ki = 520 nM T83369 CHQ5P7 118987013 Ki > 34860 nM T83369 CRI9U5 121399126 Ki = 14.8 nM T83369 CNXI35 121399185 Ki = 10.4 nM T83369 CNF2P3 121399230 Ki = 3.7 nM T83369 CPHN78 121399237 Ki = 20.8 nM T83369 C2TIC0 121399249 Ki = 3.3 nM T83369 C3F7RH 121399265 Ki = 21.8 nM T83369 CV9TX1 121399281 Ki = 9.1 nM T83369 C1ZYC9 121399296 Ki = 8 nM T83369 C4Q0HT 121399308 Ki = 15.2 nM T83369 C0G8ZE 121407232 Ki = 10.6 nM T83369 C2WD1Q 121407246 Ki = 9.8 nM T83369 C9KL5N 122192970 Ki = 19.3 nM T83369 C6SAE8 122192971 Ki = 5.7 nM T83369 CZQ6W3 122192972 Ki = 8.4 nM T83369 CX7K5B 122192988 Ki = 13.6 nM T83369 C1MVP5 122192989 Ki = 2.9 nM T83369 CLHV68 122192990 Ki = 6.2 nM T83369 CXU4S3 122193791 Ki = 12.1 nM T83369 C23NAU 122193792 Ki = 10.2 nM T83369 CX79CM 122193793 Ki = 6.9 nM T83369 C9ASN2 122193794 Ki = 5.9 nM T83369 C9Y6SO 122193795 Ki = 267.6 nM T83369 CX9T3D 122193796 Ki = 11.7 nM T83369 C2FS4M 122193797 Ki = 2.7 nM T83369 COMK61 122193798 Ki = 13.8 nM T83369 CZL3W8 122193799 Ki = 12.5 nM T83369 C90QDF 122193800 Ki = 2.1 nM T83369 CGQA72 122193881 Ki = 3 nM T83369 C9WT4R 122193882 Ki = 6.6 nM T83369 CSB1Q5 122193883 Ki = 3.1 nM T83369 C9BLF1 122193884 Ki = 4.5 nM T83369 CM0TS7 122193885 Ki = 4.2 nM T83369 CLI82V 122193886 Ki = 10.5 nM T83369 CEN5J7 122193887 Ki = 5 nM T83369 CIJ85X 122193888 Ki = 1.8 nM T83369 C13UCF 122193889 Ki = 10.5 nM T83369 CN3E4H 122193890 Ki = 34.8 nM T83369 CJS68F 122193891 Ki = 6.3 nM T83369 CTGN19 122193892 Ki = 8 nM T83369 C62TVJ 122193893 Ki = 8.4 nM T83369 CQO8Z9 122193894 Ki = 5.1 nM T83369 C9K8SJ 122193895 Ki = 1.2 nM T83369 C5R8SG 122193896 Ki = 2.4 nM T83369 C5LR2A 122193897 Ki = 2.9 nM T83369 CH2VR6 122193898 Ki = 0.8 nM T83369 CI6HC5 122193899 Ki = 2.4 nM T83369 COZP50 122193900 Ki = 1.6 nM T83369 CH46TB 122194031 Ki = 5.5 nM T83369 CGD97N 122194032 Ki = 2.6 nM T83369 C6HX9J 122194033 Ki = 0.6 nM T83369 C79TRA 122194034 Ki = 2.5 nM T83369 CN76EH 122194035 Ki = 8.6 nM T83369 CU6QD5 122194036 Ki = 0.6 nM T83369 CK0W2P 127027635 Ki > 24000 nM T83369 CPC0M8 127031390 Ki > 34860 nM T83369 CLT4P0 127032673 IC50 = 1.86 nM T83369 C8LT6S 127032674 IC50 = 11 nM T83369 CQ0Z4D 127032675 IC50 = 63.9 nM T83369 C1IL9G 135403661 Ki = 50 nM T83369 C1IGZ3 135988780 Ki = 110000 nM T83369 CK4CM2 137028369 Ki = 1 nM T83369 C7W4AS 137638513 IC50 = 2200 nM T83369 CGT80B 137640248 IC50 = 50 nM T83369 CNO2T8 137647340 IC50 > 2000000 nM T83369 C8RQW5 137647928 IC50 = 31 nM T83369 C37KPL 137648430 IC50 = 41 nM T83369 CWO52T 137653817 IC50 = 18 nM T83369 C1OXG8 137655944 IC50 = 4.9 nM T83369 CYEK02 137658233 IC50 > 3000 nM T83369 CX07YE 139592452 Ki > 27100 nM T83369 CE6C0A 145970642 Ki = 22000 nM T83369 CFJA91 145985550 Ki = 3.5 nM T83369 CICU31 155511394 Ki = 4761 nM T83369 C2VX3G 155512946 Ki > 27100 nM T83369 C2CI8S 155513907 Ki = 19724 nM T83369 CYT20V 155514020 Ki > 50000 nM T83369 CAT98N 155514640 Ki > 10000 nM T83369 C37MUL 155515203 IC50 = 36 nM T83369 CPUG37 155516479 Ki > 29000 nM T83369 CF96DM 155518671 Ki > 10000 nM T83369 C7DUX3 155520916 Ki > 10000 nM T83369 C3AL6D 155533619 IC50 = 42 nM T83369 CY3FE6 155533938 IC50 = 26 nM T83369 CL90DN 155540666 Ki > 10000 nM T83369 CU9FL4 155551858 Ki > 50000 nM T83369 CP4F1U 155567613 Ki > 50000 nM T83369 CEZ8B9 155568406 Ki > 50000 nM T83369 D03QAQ 9869498 Ki = 1900 nM T83369 D0EK9T 15230353 Ki = 1600 nM T83369 D0G4LX 46233650 Ki = 2 nM T83369 D0J1QT 44473100 Ki > 18000 nM T83369 D0JU9N 6914623 Ki > 2800 nM T83369 D0LX0D 46233193 Ki = 3800 nM T83369 D0ON2Z 204102 Ki > 2300 nM T83369 D0Y4KJ 46233192 Ki = 1900 nM T83369 D0Z2PJ 24859718 Ki = 1500 nM T13348 D09OZC 10180 IC50 = 5000 nM T13348 CI26AQ 1607 IC50 = 500 nM T13348 C5IF7O 2259 IC50 = 55 nM T13348 CHV5M7 3634 IC50 = 80 nM T13348 C6T0ZN 20477 IC50 = 50000 nM T13348 C3EOV0 51082 IC50 = 2000 nM T13348 C78ELS 67022 IC50 = 27000 nM T13348 CV75JE 76828 IC50 > 100000 nM T13348 CA5IV2 80512 IC50 = 40000 nM T13348 CP0M3Z 80695 IC50 = 8850 nM T13348 CDT53W 81409 IC50 = 3000 nM T13348 CV5EA2 94807 IC50 > 100000 nM T13348 CO52VG 104942 IC50 = 200 nM T13348 CY6VB8 107794 IC50 = 110 nM T13348 CN28KS 166754 IC50 > 100000 nM T13348 CZ58RO 223763 IC50 = 33000 nM T13348 CIQ30S 228472 IC50 = 16000 nM T13348 CN0Q4C 230714 IC50 = 1400 nM T13348 CVGN02 267570 IC50 > 200000 nM T13348 CSO78Y 322478 IC50 > 200000 nM T13348 CBF26C 329165 IC50 = 1400 nM T13348 CNSD47 356768 IC50 = 400 nM T13348 C9WI3X 460748 IC50 > 200000 nM T13348 CWYT28 460749 IC50 > 200000 nM T13348 C54MKQ 548833 IC50 = 55000 nM T13348 CU3S4G 568929 IC50 = 30000 nM T13348 CA1U0Y 580604 IC50 = 11000 nM T13348 CJLD50 646827 IC50 = 27000 nM T13348 C6TFD0 650632 IC50 = 9000 nM T13348 CE2VK6 672304 IC50 > 100000 nM T13348 C6T3MH 677363 IC50 = 15000 nM T13348 C5EF9D 677672 IC50 > 100000 nM T13348 CGE8S4 677673 IC50 = 20000 nM T13348 CSG12B 683786 IC50 = 32000 nM T13348 CGW10R 689076 IC50 = 100000 nM T13348 CZH15Y 698490 IC50 = 1500 nM T13348 CWN1Z4 702613 IC50 > 100000 nM T13348 CL15XN 707445 IC50 = 12000 nM T13348 C7UY8K 707447 IC50 = 4000 nM T13348 CAP9C2 707450 IC50 = 9000 nM T13348 C31CWM 709886 IC50 = 1600 nM T13348 CJ4Q8H 711415 IC50 > 100000 nM T13348 CSPQ54 743030 IC50 > 100000 nM T13348 CY8A4K 747735 IC50 = 33000 nM T13348 CZYE02 764976 IC50 = 30000 nM T13348 C7XMO4 766594 IC50 = 35000 nM T13348 C90MAY 768512 IC50 = 20000 nM T13348 C8X3QE 776871 IC50 = 1700 nM T13348 CH0WJ1 782036 IC50 > 100000 nM T13348 CFA26R 785306 IC50 = 20000 nM T13348 C2XID0 808751 IC50 = 100000 nM T13348 CVYL65 823651 IC50 = 6000 nM T13348 C1OEG9 823818 IC50 = 40000 nM T13348 C6WZ2C 866938 IC50 > 200000 nM T13348 CE7Y6T 873172 IC50 > 100000 nM T13348 C7WC0L 930115 IC50 > 200000 nM T13348 CJ0V3O 931081 IC50 > 200000 nM T13348 CK1TD5 941846 IC50 > 200000 nM T13348 C0ME8D 951230 IC50 > 200000 nM T13348 CB0X4T 951368 IC50 > 200000 nM T13348 CQ8D9G 1051875 IC50 > 100000 nM T13348 CAKD06 1069217 IC50 = 100000 nM T13348 C5URZ8 1080119 IC50 = 80000 nM T13348 CM7DC8 1081055 IC50 > 100000 nM T13348 C9OLR1 1087763 IC50 = 80000 nM T13348 COBH48 1092927 IC50 > 100000 nM T13348 C0PFR5 1107041 IC50 = 30000 nM T13348 CIQ94V 1117935 IC50 > 100000 nM T13348 CGX87M 1118213 IC50 > 100000 nM T13348 C5PR2L 1127114 IC50 > 100000 nM T13348 CGN76L 1127117 IC50 > 100000 nM T13348 CT80DO 1147316 IC50 > 100000 nM T13348 CV3U8A 1150481 IC50 > 100000 nM T13348 CC8U1S 1154701 IC50 > 100000 nM T13348 CQ5NX2 1177045 IC50 > 100000 nM T13348 C7JQ8I 1177061 IC50 > 100000 nM T13348 CPHF97 1202229 IC50 > 100000 nM T13348 CZRJ28 1231409 IC50 = 6000 nM T13348 CD38BH 1251742 IC50 > 100000 nM T13348 CK14MD 1270554 IC50 = 6800 nM T13348 CC2TH7 1360475 IC50 = 9000 nM T13348 CK36ZA 1428929 IC50 > 100000 nM T13348 CK62RA 1433387 IC50 > 100000 nM T13348 C7OB5V 1440680 IC50 > 100000 nM T13348 CPN73A 1441484 IC50 > 100000 nM T13348 C1R9SB 1442057 IC50 > 100000 nM T13348 COS2A9 1442144 IC50 > 100000 nM T13348 CRL81M 1452467 IC50 > 100000 nM T13348 CJ9LW5 1453572 IC50 = 40000 nM T13348 CKD60W 1460006 IC50 > 100000 nM T13348 C7G6LC 1506283 IC50 > 100000 nM T13348 C1K0NT 1582558 IC50 > 100000 nM T13348 CW59KD 1591577 IC50 > 100000 nM T13348 CJQ0B9 1594408 IC50 = 13000 nM T13348 C85TNJ 1594412 IC50 = 6000 nM T13348 C69UCE 1596134 IC50 = 50000 nM T13348 CVT65Z 1630847 IC50 = 12000 nM T13348 CIO25L 1870895 IC50 = 11000 nM T13348 C7R6VP 1889538 IC50 > 100000 nM T13348 C2FV4J 1901514 IC50 = 5000 nM T13348 C4TZ6C 1918388 IC50 = 2800 nM T13348 CI5T0N 1931499 IC50 > 100000 nM T13348 C23QYK 1963306 IC50 = 80000 nM T13348 CMPY56 1982091 IC50 = 10000 nM T13348 C5LI3R 2066037 IC50 > 100000 nM T13348 C1SZC8 2178259 IC50 = 17000 nM T13348 CG6UJ4 2256566 IC50 = 6000 nM T13348 CPW47J 2274649 IC50 > 100000 nM T13348 CH8AJ0 2392662 IC50 = 3000 nM T13348 C5V6MG 2718237 IC50 > 100000 nM T13348 CMU3O8 2731081 IC50 = 2000 nM T13348 C1WE9N 2741156 IC50 = 1300 nM T13348 CY0N8W 2772235 IC50 > 100000 nM T13348 C27PJX 2772535 IC50 = 4000 nM T13348 CSTG29 2772554 IC50 = 19000 nM T13348 CB42CF 2784232 IC50 > 100000 nM T13348 C94DXQ 2798966 IC50 = 1800 nM T13348 CM27NB 2802503 IC50 > 100000 nM T13348 CYUD59 2828740 IC50 = 40000 nM T13348 CHYJ43 2835401 IC50 = 6000 nM T13348 C9B4DK 2856194 IC50 = 100000 nM T13348 C2SHI8 2859804 IC50 = 16000 nM T13348 CWTP79 2866638 IC50 > 100000 nM T13348 CYJ59S 2868785 IC50 = 11000 nM T13348 CK73ZP 2872940 IC50 = 3000 nM T13348 CLE4N8 2876082 IC50 > 100000 nM T13348 C0TG1R 2947382 IC50 > 100000 nM T13348 C1VB6G 2959829 IC50 > 100000 nM T13348 C2H1YR 2997176 IC50 > 100000 nM T13348 C71CWL 2997361 IC50 > 100000 nM T13348 C14JGA 3090411 IC50 = 35000 nM T13348 CM2R3O 3092313 IC50 = 8000 nM T13348 C0D3QT 3107546 IC50 > 100000 nM T13348 CSN8Y1 3109045 IC50 = 60000 nM T13348 CU25JK 3111071 IC50 = 100000 nM T13348 C3L8ED 3111089 IC50 > 100000 nM T13348 CRD48U 3113864 IC50 > 100000 nM T13348 C4XRO3 3115317 IC50 > 100000 nM T13348 CM3LG7 3121209 IC50 = 8000 nM T13348 C67VFW 3127906 IC50 > 100000 nM T13348 C7C1EL 3130462 IC50 > 100000 nM T13348 C7OPF8 3130858 IC50 = 50000 nM T13348 CA62JR 3131586 IC50 = 40000 nM T13348 CMG97N 3134919 IC50 = 27000 nM T13348 CZ9KQ0 3134995 IC50 > 100000 nM T13348 CWY0L7 3137464 IC50 > 100000 nM T13348 CK7DN2 3137465 IC50 > 100000 nM T13348 C8PD5T 3149147 IC50 = 80000 nM T13348 CQ9FS3 3150744 IC50 > 100000 nM T13348 C9E0DK 3153711 IC50 > 100000 nM T13348 C02AOL 3155633 IC50 = 26000 nM T13348 C8AS6J 3155998 IC50 > 100000 nM T13348 CHQ64T 3158634 IC50 > 100000 nM T13348 C89AVP 3159575 IC50 > 100000 nM T13348 C35DCU 3164059 IC50 > 200000 nM T13348 CNTJ89 3164066 IC50 > 200000 nM T13348 CSXC46 3164070 IC50 > 200000 nM T13348 CM31FX 3164796 IC50 > 100000 nM T13348 C1DP7F 3167551 IC50 > 100000 nM T13348 CJ7KO2 3168504 IC50 > 100000 nM T13348 C1OCF8 3169644 IC50 > 100000 nM T13348 C6Y2VD 3173689 IC50 > 100000 nM T13348 CN52TE 3177833 IC50 > 100000 nM T13348 CZA37W 3181074 IC50 > 100000 nM T13348 CS1A9O 3184366 IC50 > 100000 nM T13348 C3O1RA 3189845 IC50 > 100000 nM T13348 CH6RJ0 3191968 IC50 > 100000 nM T13348 C3GUM6 3202192 IC50 > 100000 nM T13348 CA7EJ4 3206523 IC50 > 100000 nM T13348 CY6T7O 3219677 IC50 > 100000 nM T13348 CE12BS 3225890 IC50 > 100000 nM T13348 CU81OI 3225961 IC50 > 100000 nM T13348 C0R9IX 3227536 IC50 > 100000 nM T13348 CKLA53 3232099 IC50 > 100000 nM T13348 CDN2X1 3239254 IC50 = 7070 nM T13348 CJ3V0P 3246032 IC50 = 1700 nM T13348 C1SZT4 3431959 IC50 = 4000 nM T13348 CE9Z1H 3581333 IC50 = 12000 nM T13348 CH92NQ 3638737 IC50 = 250 nM T13348 CP0ZA7 4055306 IC50 = 3800 nM T13348 CN2C4Z 4177223 IC50 = 6800 nM T13348 CF1NQ0 4275874 IC50 = 8300 nM T13348 CKCY57 4981199 IC50 = 800 nM T13348 C2C9RE 4989139 IC50 > 200000 nM T13348 CY1NB7 5075788 IC50 = 1600 nM T13348 CAT76G 5306626 IC50 > 100000 nM T13348 CG2V7P 5708138 IC50 > 100000 nM T13348 CO8M4Q 6411132 IC50 > 200000 nM T13348 CGCJ60 6439397 IC50 = 10000 nM T13348 C2BY6K 6458554 IC50 > 200000 nM T13348 CVC31J 6459022 IC50 > 200000 nM T13348 CK67QL 6462917 IC50 > 100000 nM T13348 CE92LT 6486669 IC50 > 100000 nM T13348 CTA32I 6489396 IC50 > 100000 nM T13348 C85CMY 6491348 IC50 > 100000 nM T13348 C5WY1S 6492340 IC50 > 100000 nM T13348 C3PO7W 6493581 IC50 = 100000 nM T13348 CC6U7A 6493950 IC50 > 200000 nM T13348 C94EOZ 6494960 IC50 > 100000 nM T13348 C2ZLP7 6495034 IC50 > 100000 nM T13348 CD3JG9 6495052 IC50 > 100000 nM T13348 CE1K8O 6496782 IC50 > 100000 nM T13348 C25KZS 6501515 IC50 > 100000 nM T13348 CPR2D1 6502965 IC50 > 100000 nM T13348 COVE16 6503001 IC50 > 100000 nM T13348 C5OT9B 6604161 IC50 = 250 nM T13348 CEN4Z3 6710858 IC50 = 900 nM T13348 C7UD2S 9555458 IC50 = 2900 nM T13348 CM95CS 9555464 IC50 = 4100 nM T13348 CGQC13 9555467 IC50 = 4400 nM T13348 C7NFC3 13518539 IC50 = 40000 nM T13348 C8Z9XB 16481078 IC50 > 200000 nM T13348 C8YE0J 25190436 IC50 = 15000 nM T13348 CLK32U 25190437 IC50 = 22000 nM T13348 CO9PA5 25190438 IC50 = 6000 nM T13348 C6ZA4E 25210558 IC50 = 1000 nM T13348 CZEB56 25235419 IC50 = 3000 nM T13348 CU3I5T 25235420 IC50 = 3000 nM T13348 C5TQ3U 25235421 IC50 = 15000 nM T13348 CO0AP7 25235422 IC50 = 10000 nM T13348 CT6RZ4 25235423 IC50 = 3000 nM T13348 COLK18 25235424 IC50 = 15000 nM T13348 C3BI5U 25235425 IC50 = 4000 nM T13348 C2ZHV4 25235426 IC50 = 1000 nM T13348 C1VZA5 25235467 IC50 = 2000 nM T13348 CBI08X 25235468 IC50 = 1000 nM T13348 C0S1MF 25235469 IC50 = 1000 nM T13348 C7QM0X 25235471 IC50 = 10000 nM T13348 CB78PF 25235472 IC50 = 1000 nM T13348 C65HIF 44569337 IC50 > 100000 nM T13348 CX6FE2 44569348 IC50 = 4000 nM T13348 CJ58ZM 44569595 IC50 > 100000 nM T13348 C93CUT 45266435 IC50 > 100000 nM T13348 C5YL2E 45487238 IC50 = 10000 nM T13348 C2WP9E 45487270 IC50 = 2000 nM T13348 CKZR30 45487277 IC50 = 3000 nM T13348 CFBT48 46833159 IC50 > 200000 nM T13348 COS86H 46834048 IC50 > 200000 nM T13348 CV60DR 46834317 IC50 > 200000 nM T13348 C05YOF 46925861 IC50 = 4000 nM T13348 CZM45N 46925862 IC50 = 11100 nM T13348 C1O5SA 46925863 IC50 > 57000 nM T13348 C5NXV8 46925867 IC50 = 17600 nM T13348 CZ61HG 46925868 IC50 = 18200 nM T13348 C9QZC3 46925869 IC50 = 12000 nM T13348 CG40SU 46925870 IC50 = 13000 nM T13348 C5V7EZ 46925871 IC50 > 57000 nM T13348 CNJ76F 46925873 IC50 > 57000 nM T13348 CS0D2V 46925875 IC50 = 3100 nM T13348 C7IQY9 46925876 IC50 > 57000 nM T13348 CLJ2P5 46925877 IC50 = 19000 nM T13348 CWY1M6 46925878 IC50 = 25200 nM T13348 CUZ85I 46925879 IC50 = 2900 nM T13348 CA43PG 46925884 IC50 = 1000 nM T13348 CGA4T5 46925885 IC50 = 2900 nM T13348 CP50XO 46925888 IC50 = 13000 nM T13348 CCA6Z3 46925889 IC50 = 14000 nM T13348 C1QOG5 49852733 IC50 > 57000 nM T13348 CHK54A 49852899 IC50 > 57000 nM T13348 C1NTC4 49852971 IC50 > 57000 nM T13348 CZY43Q 49853107 IC50 > 57000 nM T13348 CC1ZE2 49853161 IC50 = 9100 nM T13348 CG0F1E 49853292 IC50 = 5300 nM T13348 C2SEN9 49853346 IC50 > 57000 nM T13348 COR8H3 57387292 IC50 > 57000 nM T13348 C9KSB1 57387550 IC50 = 6000 nM T13348 CP14ZD 57387552 IC50 > 57000 nM T13348 C3UI9S 70676765 IC50 = 19000 nM T13348 C1HKR2 70676766 IC50 = 18000 nM T13348 C5TWX8 70676768 IC50 = 16000 nM T13348 CRV07P 70676769 IC50 = 18000 nM T13348 CA1EI3 70701319 IC50 = 55 nM T13348 C8VRI9 71479367 IC50 = 8500 nM T13348 CU8ZA0 71817697 IC50 > 200000 nM T13348 CLD4B7 71817698 IC50 > 200000 nM T13348 CZE8Q2 71817849 IC50 > 200000 nM T13348 CG2A6C 71817850 IC50 > 200000 nM T13348 C2ZYW4 71817852 IC50 > 200000 nM T13348 C35QBR 71817853 IC50 > 200000 nM T13348 C8A0CS 71818002 IC50 > 200000 nM T13348 CHKS75 71818003 IC50 > 200000 nM T13348 CJ3YG9 71818004 IC50 > 200000 nM T13348 C8WN0H 71818005 IC50 > 200000 nM T13348 C4HGP6 71818006 IC50 > 200000 nM T13348 CEX8A6 71818007 IC50 > 200000 nM T13348 CPB21Q 71818143 IC50 > 200000 nM T13348 CTD4U6 71818144 IC50 > 200000 nM T13348 C7UB6O 71818145 IC50 > 200000 nM T13348 CHF45Y 71818146 IC50 > 200000 nM T13348 C96AYZ 71818147 IC50 > 200000 nM T13348 CJ2OV6 71818149 IC50 > 200000 nM T13348 CLAF94 71818291 IC50 > 200000 nM T13348 CWHG19 71818293 IC50 > 200000 nM T13348 CH6BV1 71818296 IC50 > 200000 nM T13348 CHN47D 71818443 IC50 > 200000 nM T13348 CZXW74 71818444 IC50 > 200000 nM T13348 C7TIJ1 71818716 IC50 > 200000 nM T13348 CLU15O 71818717 IC50 > 200000 nM T13348 CF9I3P 71818718 IC50 > 200000 nM T13348 C3DTB4 71818719 IC50 > 200000 nM T13348 CI80ND 71818720 IC50 > 200000 nM T13348 COU9C7 71818721 IC50 > 200000 nM T13348 C8AR0I 71818722 IC50 > 200000 nM T13348 CB23IX 71818723 IC50 > 200000 nM T13348 CQV2B5 71818864 IC50 > 200000 nM T13348 C8L1XF 71818865 IC50 > 200000 nM T13348 C5CXH0 71818866 IC50 > 200000 nM T13348 C7P2XN 71818867 IC50 > 200000 nM T13348 CPK26T 71818868 IC50 > 200000 nM T13348 C85OTM 71818869 IC50 > 200000 nM T13348 CK6W2Z 71818870 IC50 > 200000 nM T13348 C9MKT5 71819004 IC50 > 200000 nM T13348 CMI5O8 71819005 IC50 > 200000 nM T13348 CG7ZN2 71819006 IC50 > 200000 nM T13348 CWSE58 71819007 IC50 > 200000 nM T13348 CXG20Y 71819008 IC50 > 200000 nM T13348 CMT0Y2 71819009 IC50 > 200000 nM T13348 C48DOI 71819143 IC50 > 200000 nM T13348 CJC48A 71819144 IC50 > 200000 nM T13348 C7GXZ3 71819145 IC50 > 200000 nM T13348 C7Q0NF 71819146 IC50 > 200000 nM T13348 C5ET9H 71819147 IC50 > 200000 nM T13348 CRZ8G6 71819148 IC50 > 200000 nM T13348 C19SNE 71819283 IC50 > 200000 nM T13348 C6NQP9 73346151 IC50 > 200000 nM T13348 C9CI3X 73350770 IC50 > 200000 nM T13348 C52BOT 73441016 IC50 = 2500 nM T13348 CF59JM 135427565 IC50 = 87000 nM T13348 C41BEK 135452745 IC50 > 100000 nM T13348 C42RHY 135457569 IC50 > 100000 nM T13348 C32VMB 135464628 IC50 = 50000 nM T13348 CV7AF2 135470272 IC50 > 100000 nM T13348 C0RO8W 135477708 IC50 = 33000 nM T13348 C0U8KB 135477719 IC50 > 100000 nM T13348 CHP0Z8 135477753 IC50 > 100000 nM T13348 CM28FI 135483971 IC50 = 400 nM T13348 C8F3AZ 135495851 IC50 > 100000 nM T13348 C6ERF8 135764771 IC50 = 7760 nM T13348 CRG3L9 145967342 IC50 = 1800 nM T13348 CZXB86 145967413 IC50 = 2000 nM T13348 CGN3H5 145975142 IC50 = 57 nM T13348 CLH26X 145976435 IC50 = 1700 nM T13348 C0EYP1 145978323 IC50 = 250 nM T13348 CBO26Z 155512913 IC50 = 33200 nM T13348 CZV47T 155525162 IC50 = 5700 nM T13348 CR85AP 155525896 IC50 = 29200 nM T13348 C40FDX 155527118 IC50 = 1800 nM T13348 CB5MP2 155528025 IC50 = 2700 nM T13348 CPH2M4 155530918 IC50 = 2600 nM T13348 CMK3G6 155531117 IC50 = 2500 nM T13348 CJTN37 155536398 IC50 = 1300 nM T13348 C1D6QJ 155536768 IC50 > 50000 nM T13348 C2TMZ8 155537771 IC50 > 100000 nM T13348 CVIP75 155539397 IC50 = 26500 nM T13348 COS0U2 155541086 IC50 = 1200 nM T13348 CAV1O3 155546896 IC50 = 55100 nM T13348 COU2R3 155549369 IC50 = 9300 nM T13348 CEC7I9 155549877 IC50 = 12100 nM T13348 CE06MB 155553113 IC50 = 63500 nM T13348 C9ZW4T 155553528 IC50 > 100000 nM T13348 CL28QD 155555676 IC50 = 10600 nM T13348 CUM47N 155556285 IC50 = 52600 nM T13348 C4T1FJ 155560911 IC50 = 5400 nM T13348 CS2O3W 155561453 IC50 = 1900 nM T13348 D07DZS 1240423 IC50 = 3000 nM T13348 D0NH7M 5328760 IC50 = 280 nM T13348 D0P0CM 460747 IC50 > 200000 nM T13348 D0T3PW 5281672 IC50 = 320 nM T79798 D0EG1I 9926791 IC50 > 10000 nM T79798 D03LWG 53235510 IC50 > 10000 nM T79798 D07EHV 44814409 IC50 > 10000 nM T79798 D0A5HC 45109868 IC50 = 40 nM T79798 D0E3TC 44259 IC50 = 275 nM T79798 D0O6ZO 9952773 IC50 > 10000 nM T79798 D0T3ME 156422 IC50 = 30 nM T79798 CL5I2U 5330279 IC50 > 10000 nM T79798 C20RSC 9811100 IC50 > 10000 nM T79798 CJO47T 9948405 IC50 > 10000 nM T79798 CV8I5X 9999342 IC50 > 10000 nM T79798 C7YD1X 10048045 IC50 > 25000 nM T79798 CCE2T5 10229750 IC50 = 213 nM T79798 C5TQ7X 10247543 IC50 > 10000 nM T79798 CV1WZ5 10301047 IC50 = 2050 nM T79798 C2WQ8M 10473563 IC50 > 10000 nM T79798 COE34F 11103319 IC50 = 616 nM T79798 C2W5RC 11235063 IC50 > 30000 nM T79798 CBOP58 11293798 Ki > 10000 nM T79798 C26BZX 11362471 Ki > 10000 nM T79798 CWXB93 11397177 Ki > 10000 nM T79798 C71PYD 11427975 IC50 > 30000 nM T79798 CTG83F 11539329 Ki > 7500 nM T79798 CACS26 11561968 Ki > 2000 nM T79798 CMIL86 11590363 Ki > 7500 nM T79798 C9T6SC 11640926 Ki > 7500 nM T79798 CU0E8O 11690457 Ki > 2000 nM T79798 CFPW41 16007116 Ki > 7500 nM T79798 C9TU1O 16046126 IC50 > 1000 nM T79798 C75DWA 23400208 IC50 > 30000 nM T79798 CG6D4M 23647319 IC50 > 10000 nM T79798 CY8Z7X 23647330 IC50 > 10000 nM T79798 C4XD8H 23647348 IC50 > 10000 nM T79798 CY8L7E 24896769 IC50 > 10000 nM T79798 CVQS96 25052767 Ki = 3500 nM T79798 CU80BP 44517743 IC50 > 10000 nM T79798 C5Z3LI 44591740 IC50 = 6200 nM T79798 CVED60 45254198 IC50 = 461 nM T79798 C53MQJ 45254575 IC50 = 647 nM T79798 CS9Y8K 45254577 IC50 = 169 nM T79798 C7YCA2 45257074 IC50 = 148 nM T79798 C19HUI 45257075 IC50 = 352 nM T79798 CY3HW5 46224684 IC50 = 4000 nM T79798 C2P9QO 46228508 IC50 = 1810 nM T79798 C6E5PY 46228822 IC50 > 10000 nM T79798 C3T8AM 46228951 IC50 > 10000 nM T79798 CX8MJ9 46836027 IC50 = 354 nM T79798 CS8NX0 46836043 IC50 = 902 nM T79798 CLS29B 46872626 IC50 > 10000 nM T79798 C2O8RZ 46886323 IC50 > 1000 nM T79798 CHSF07 49806372 IC50 > 1000 nM T79798 C6DC4S 53241447 IC50 = 55 nM T79798 C8NA4L 53384644 IC50 > 30000 nM T79798 CP1FH5 53391990 IC50 = 195 nM T79798 C4JCT1 53476174 IC50 = 972 nM T79798 C1XS2J 54760383 IC50 > 10000 nM T79798 C6HR5F 58416745 IC50 = 1504 nM T79798 CRY9K7 58416748 IC50 = 591 nM T79798 CYI32L 58532548 IC50 = 1941 nM T79798 C1MR8Q 60097495 IC50 > 10000 nM T79798 CV63UL 67240318 IC50 > 10000 nM T79798 C3NHU5 127030449 IC50 = 634 nM T79798 CI73JH 127030772 IC50 > 17000 nM T79798 CEI25F 127030791 IC50 > 17000 nM T79798 CUQ5T4 127030792 IC50 = 303 nM T79798 C7Q6PH 127030793 IC50 = 8359 nM T79798 CRO3B9 127031107 IC50 > 16000 nM T79798 CXV6F2 127031108 IC50 > 15000 nM T79798 C90LYU 127031109 IC50 > 17000 nM T79798 CD5A9R 127031117 IC50 = 378 nM T79798 CV7KB9 127031414 IC50 > 16000 nM T79798 CANH59 127031725 IC50 = 2438 nM T79798 C3UDF1 127034594 IC50 = 2950 nM T79798 C6VB3O 145925651 IC50 >= 5000 nM T79798 C2MD1Q 155513187 IC50 > 10000 nM T79798 D00ERW 44444843 Ki > 7500 nM T79798 D00HVA 11624601 Ki > 7500 nM T79798 D08LYB 5166 IC50 > 100000 nM T79798 D0C7RS 1369 IC50 > 40000 nM T79798 D0Q3NG 11715520 Ki > 7500 nM T79798 D0S7IE 11658882 Ki > 7500 nM T73134 D0MU9L 176077 IC50 = 90000 nM T73134 CCFH71 11313 IC50 = 100000 nM T73134 C9Z3SR 17341 IC50 = 600000 nM T73134 C6WXE2 19098 IC50 = 600000 nM T73134 CXEC70 69439 IC50 = 80000 nM T73134 CUJ90R 75195 IC50 = 200000 nM T73134 C7RJ0Z 200980 IC50 = 90000 nM T73134 CHY93K 447607 IC50 > 10000 nM T73134 CIPB41 480947 Ki = 72000 nM T73134 CK9N7A 513282 Ki = 6400 nM T73134 CG8D0N 513283 Ki = 13000 nM T73134 C03SRB 513284 IC50 = 500000 nM T73134 CDB17F 1538822 IC50 = 55000 nM T73134 C4KO1Z 2799782 IC50 = 15000 nM T73134 CR3NG2 5190983 IC50 = 320000 nM T73134 CJ6TV8 10011928 IC50 > 1000000 nM T73134 COC14Z 10039700 IC50 = 125 nM T73134 CE9XP3 10240946 IC50 = 240 nM T73134 CP42KR 11029971 IC50 = 600000 nM T73134 CT3R7M 11580364 Ki = 330000 nM T73134 C59WNV 13329882 IC50 = 720000 nM T73134 CRLD46 44292607 IC50 = 150000 nM T73134 CYBM80 44367875 IC50 > 1000000 nM T73134 CF7H4C 44368231 IC50 > 1000000 nM T73134 C75BDZ 44368232 IC50 > 1000000 nM T73134 CS5ZN1 44368239 IC50 = 43000 nM T73134 C7UOE9 44410200 Ki = 300 nM T73134 C8NK5J 44461886 Ki = 25000 nM T73134 CR58OQ 44563274 Ki = 700 nM T73134 CLA85J 44563275 Ki = 600 nM T73134 C7NJ6K 52912443 IC50 = 3000 nM T73134 CZ4Y7R 53358441 Ki = 700 nM T73134 CWPA60 71573724 IC50 = 46000 nM T73134 C5W3CM 101735280 IC50 = 250 nM T73134 CLPT86 122657813 IC50 = 10 nM T73134 CB90TF 122657820 IC50 = 0.4 nM T73134 C30RWL 127027504 IC50 = 2420 nM T73134 C9J8LD 127027505 IC50 = 210 nM T73134 CD0IP7 127034618 IC50 = 43000 nM T73134 C76JWP 127034620 IC50 > 1000000 nM T73134 CAF9D8 127034622 IC50 = 41000 nM T73134 C1GX2A 127034624 IC50 = 15000 nM T73134 CG0M8L 127034626 IC50 = 60000 nM T73134 C1KA0S 127034628 IC50 = 490000 nM T73134 CWDC64 127034630 IC50 = 28000 nM T73134 CV03JM 127034632 IC50 = 86000 nM T73134 CHY10W 127035143 IC50 = 50000 nM T73134 CO3R1K 127035145 IC50 = 19000 nM T73134 CLSC85 127035326 IC50 > 1000000 nM T73134 CO52UV 127035677 IC50 = 56000 nM T73134 C5S0JI 127036664 IC50 = 180000 nM T73134 CW2DX5 127037636 IC50 = 120000 nM T73134 C5U4IT 135576411 IC50 = 180000 nM T73134 CQT81G 137640259 Ki = 290 nM T73134 C2FY5W 137644530 Ki = 9200 nM T73134 C9NFJ1 137645268 IC50 > 150000 nM T73134 CM6G4Y 137661178 IC50 = 13000 nM T73134 COEN10 145991014 IC50 = 10 nM T73134 D0R8TR 445612 IC50 = 40000 nM T86829 CUBE62 449402 Ki = 0.03 nM T86829 CXZ13O 449484 Ki = 0.008 nM T86829 C8YNF2 800130 Ki = 520 nM T86829 CQT58L 5496910 Ki = 0.046 nM T86829 CC0BA1 5496989 Ki = 0.032 nM T86829 CWQZ70 11527333 Ki = 0.036 nM T86829 CY1KM5 19094087 Ki = 45000 nM T86829 C70KPI 23446862 Ki = 0.03 nM T86829 CM96ZQ 23550313 Ki = 0.016 nM T86829 C9F5MR 23550315 Ki = 0.012 nM T86829 C7QVW9 23550316 Ki = 0.42 nM T86829 CQN03W 23550318 Ki = 0.35 nM T86829 CXF2S6 23550321 Ki = 0.1 nM T86829 C2JWB1 23550322 Ki = 0.016 nM T86829 CR70HT 23550323 Ki = 0.026 nM T86829 C73GNY 23550324 Ki = 0.011 nM T86829 C3U1TN 23550325 Ki = 0.067 nM T86829 CA1P5N 44288152 Ki = 66 nM T86829 CY97ZS 44288153 Ki = 0.58 nM T86829 C1SG7L 44288172 Ki = 0.014 nM T86829 C9IT4Y 44288173 Ki = 0.02 nM T86829 C7P4TR 44288207 Ki = 7.7 nM T86829 C1G3QB 44288209 Ki = 0.042 nM T86829 C6OC4V 44288228 Ki = 0.02 nM T86829 CZNS25 44288229 Ki = 0.02 nM T86829 CW2FO8 44288248 Ki = 33 nM T86829 CY6LC3 44288269 Ki = 0.07 nM T86829 CI5K1O 44288279 Ki = 0.38 nM T86829 CKS5X9 44288280 Ki = 7.5 nM T86829 CY4RV8 44288283 Ki = 0.085 nM T86829 CBN0S2 44288298 Ki = 0.08 nM T86829 CSY43L 44288299 Ki = 1.7 nM T86829 C98JHL 44288300 Ki = 2.2 nM T86829 CG28KN 44288325 Ki = 0.021 nM T86829 CZCQ23 44288326 Ki = 0.27 nM T86829 C2TQ5R 44288454 Ki = 0.076 nM T86829 CBH74P 44288459 Ki = 13.6 nM T86829 C81XHJ 44288516 Ki = 2.8 nM T86829 CME72B 44288540 Ki = 7.2 nM T86829 C4KYO7 44288550 Ki = 0.14 nM T86829 C73DRB 44288559 Ki = 0.034 nM T86829 CO3B1Y 44288577 Ki = 0.038 nM T86829 C9SE1N 44288599 Ki = 97 nM T86829 CBC81Z 44288604 Ki = 5.5 nM T86829 C1B8OH 44288642 Ki = 0.95 nM T86829 C7SYO4 44288643 Ki = 0.24 nM T86829 CNAC20 44288644 Ki = 0.46 nM T86829 C5QCS1 44288645 Ki = 0.034 nM T86829 CJ20RU 44288646 Ki = 0.019 nM T86829 C0NLM7 44288667 Ki = 0.24 nM T86829 COM87L 44288668 Ki = 0.44 nM T86829 CB98AM 44288671 Ki = 0.83 nM T86829 CDC2U9 44288674 Ki = 0.031 nM T86829 CVGF63 44288676 Ki = 1.1 nM T86829 CPWD59 44288692 Ki = 1.9 nM T86829 C9Z3JY 44288748 Ki = 0.11 nM T86829 C9G5DB 44288750 Ki = 0.17 nM T86829 C9GV3R 44288762 Ki = 0.37 nM T86829 CI6B8P 44288763 Ki = 0.22 nM T86829 CH87BC 44318364 Ki = 5.6 nM T86829 CW4U1P 44318393 Ki = 8.6 nM T86829 C4ETC5 44364141 Ki = 6.4 nM T86829 CJC84Z 54457761 Ki = 0.45 nM T86829 CF7E6V 69117064 Ki = 0.13 nM T86829 CP63UY 69471397 Ki = 6 nM T86829 C7XR1O 76308260 Ki = 16 nM T86829 C34MGR 76308261 Ki = 28 nM T86829 CN36WV 76319133 Ki = 3.2 nM T86829 CKZ86Y 76319134 Ki = 3.2 nM T86829 CYI68H 76322794 Ki = 0.31 nM T86829 CJ62LA 76322795 Ki = 0.021 nM T86829 C6B8EC 76326355 Ki = 0.057 nM T86829 CTZ0J5 76329966 Ki = 44 nM T86829 D05OPY 44288306 Ki = 19 nM T86829 D07CEB 44288035 Ki = 2300 nM T86829 D09XXN 2287872 Ki = 7.3 nM T62276 CB50FH 6604872 IC50 = 5 nM T62276 CWP9R2 9799046 IC50 = 2 nM T62276 C7JAZ2 9863010 IC50 = 35000 nM T62276 C1OY3T 9863759 IC50 = 1 nM T62276 CC56WK 9998801 IC50 = 8.2 nM T62276 CB8KW6 10048025 IC50 = 8 nM T62276 C7RTW2 10498624 IC50 = 52000 nM T62276 C8HVN0 10547776 IC50 = 19 nM T62276 CKG69I 10569480 IC50 = 110 nM T62276 CR69GF 10594749 IC50 = 19 nM T62276 CGQ14N 10618608 IC50 = 25000 nM T62276 C73NYU 10640029 IC50 = 15000 nM T62276 C1S4WZ 10640185 IC50 = 420 nM T62276 CFP76T 10688762 IC50 = 250 nM T62276 C2YE1S 10689828 IC50 = 17 nM T62276 CWO6V0 10736249 IC50 = 220 nM T62276 C09CWU 10737190 IC50 > 100000 nM T62276 CWF96L 10738253 IC50 = 180 nM T62276 CQJ2T4 10758743 IC50 = 380 nM T62276 C8JT1X 10760940 IC50 = 62000 nM T62276 CGJ1W6 10761824 IC50 = 57000 nM T62276 CBO3A8 10783792 IC50 = 49 nM T62276 C5W2NG 10784705 IC50 = 89 nM T62276 C9V0FI 10808704 IC50 = 6.1 nM T62276 C6SMO8 10809420 IC50 = 1100 nM T62276 C62RYJ 10809482 IC50 = 26 nM T62276 C12GHB 10832383 IC50 = 120 nM T62276 CSP5G0 10960335 Ki = 990 nM T62276 CJD9A5 11014327 Ki = 14 nM T62276 C8OW0I 11035463 Ki = 92000 nM T62276 C4Z9LY 11046684 Ki = 120 nM T62276 CV8MJ5 11079958 Ki = 58 nM T62276 C9OCK4 11091488 Ki = 72 nM T62276 C6JF8W 17878056 IC50 = 40 nM T62276 CN2M7T 22096990 IC50 = 2 nM T62276 CD8YQ1 23661726 IC50 = 27 nM T62276 C2J7HX 44318983 IC50 = 32 nM T62276 C5PY4M 44319073 IC50 = 8 nM T62276 C9L1NA 44378229 IC50 = 76 nM T62276 CB9FS4 44378279 IC50 = 9 nM T62276 CO49DT 44378434 IC50 = 6 nM T62276 C6CY2O 44443053 IC50 = 14 nM T62276 C9SLD8 44443054 IC50 = 4 nM T62276 C71NKB 44443055 IC50 = 58 nM T62276 C3OA0D 44443059 IC50 = 41 nM T62276 CG01OQ 44443061 IC50 = 12 nM T62276 C9D3YS 44443062 IC50 = 45 nM T62276 C43XEC 44443064 IC50 = 39 nM T62276 CYBX43 44443065 IC50 = 59 nM T62276 CY36XN 44443066 IC50 = 166 nM T62276 CLXD29 44443067 IC50 = 38 nM T62276 CZ82GA 44443069 IC50 = 8 nM T62276 CX5F7M 44443071 IC50 = 209 nM T62276 CG16MU 44443072 IC50 = 19 nM T62276 CM18FN 44443073 IC50 = 11 nM T62276 CDW01E 44443074 IC50 = 728 nM T62276 C67TZR 44443075 IC50 = 77 nM T62276 C4LMB6 44443077 IC50 = 74 nM T62276 CU8A3F 44443078 IC50 = 49 nM T62276 D03GBO 127988 Ki = 2900 nM T15745 CZI4N9 13387 IC50 = 34000000 nM T15745 C72LED 82316 IC50 = 826000 nM T15745 CQ43EI 648697 IC50 = 37000 nM T15745 CG84JK 709639 IC50 = 26000 nM T15745 CTX78N 1268265 IC50 = 279000 nM T15745 C2M0SE 1511198 IC50 > 100000 nM T15745 CJK1F0 1511199 IC50 > 100000 nM T15745 CE23CA 2780190 IC50 = 476000 nM T15745 CDQ74H 2796714 IC50 = 495000 nM T15745 C0CG1E 2797467 IC50 = 190000 nM T15745 CR3SF5 4907545 IC50 > 100000 nM T15745 CWG19Q 4908238 IC50 > 100000 nM T15745 CF48PO 19279808 IC50 = 1094000 nM T15745 CI6LM0 24229802 IC50 = 109000 nM T15745 CD3X6J 24229806 IC50 = 241000 nM T15745 CA9X1J 24229807 IC50 = 38000 nM T15745 C61JHB 29133832 IC50 = 37000 nM T15745 CUF8V6 29147548 IC50 = 36000 nM T15745 CWH6I9 32854678 IC50 = 12000 nM T15745 CRD38P 42582730 IC50 = 102000 nM T15745 CY86UV 47306828 IC50 = 9000 nM T15745 CG3PR6 52912222 IC50 > 31622.78 nM T15745 C1KWY4 54759170 IC50 = 7000 nM T15745 CUZR69 70680607 IC50 = 3162.28 nM T15745 CM90YZ 70680608 IC50 = 610 nM T15745 CDY89S 70680609 IC50 = 840 nM T15745 CIPN50 71760902 IC50 > 1000 nM T15745 C2ZW4L 76310337 IC50 > 2000000 nM T15745 C1E3NI 76310338 IC50 = 143000 nM T15745 CZK7V3 76314006 IC50 = 69000 nM T15745 CZCR56 76317546 IC50 = 25000 nM T15745 CEJ36W 76317548 IC50 = 55000 nM T15745 CL5O0E 76317549 IC50 > 1000000 nM T15745 CFQG10 76321282 IC50 = 152000 nM T15745 C6JRU2 76321284 IC50 = 46000 nM T15745 C59WEA 76324896 IC50 = 66000 nM T15745 C5TW8D 76324897 IC50 = 50000 nM T15745 C9HXI6 76335752 IC50 = 37000 nM T15745 CQ0IP7 76335754 IC50 = 14000 nM T15745 C5TB9S 77843982 IC50 > 1000 nM T15745 CJQ9Z5 91971269 IC50 = 27000 nM T15745 C9WB3G 95828281 IC50 > 20000 nM T15745 C8BMH6 118733097 IC50 = 4400 nM T15745 CTD04M 118733098 IC50 > 50000 nM T15745 CUF52T 118733099 IC50 = 5250 nM T15745 CQ7ZG2 118733100 IC50 > 50000 nM T15745 C3Y2KO 118733101 IC50 > 50000 nM T15745 CYTV76 118733102 IC50 > 50000 nM T15745 C8A2IN 118733103 IC50 = 770 nM T15745 C2BO5U 118733104 IC50 = 790 nM T15745 C7Q0IC 118733105 IC50 = 2450 nM T15745 CUWX94 119081692 IC50 = 3600 nM T15745 CDH8M4 121373418 IC50 > 20000 nM T15745 C47QXT 121376807 IC50 > 20000 nM T15745 C15SUJ 127025079 IC50 = 9800 nM T15745 CMG7C1 127026579 IC50 = 1000 nM T15745 CAV92O 127026580 IC50 = 4100 nM T15745 C9WLR6 127026581 IC50 = 3800 nM T15745 C57IHP 127026582 IC50 = 1300 nM T15745 CM97ZL 127026583 IC50 = 370 nM T15745 C7WE5X 127026588 IC50 = 410 nM T15745 CB2CX8 127026589 IC50 = 540 nM T15745 CRFG40 127026590 IC50 = 1900 nM T15745 CF9QV5 127026591 IC50 = 820 nM T15745 C6GR7I 127026628 IC50 > 30000 nM T15745 CY7T5G 127026629 IC50 = 22700 nM T15745 C3LM6B 127026630 IC50 = 12500 nM T15745 C35AYZ 127027784 IC50 = 1900 nM T15745 CXL45V 127028085 IC50 = 1500 nM T15745 C0C1HZ 127028091 IC50 = 670 nM T15745 CAH3Q7 127029580 IC50 = 34100 nM T15745 C3R8FQ 127038798 IC50 > 100000 nM T15745 CBNZ13 127040778 IC50 = 2511.89 nM T15745 CTA9I1 127042046 IC50 = 15848.93 nM T15745 CWVS97 127043088 IC50 = 8550 nM T15745 CGDN94 132275066 IC50 > 18000 nM T15745 CU2F1G 135566900 Ki = 2260 nM T15745 CW94QO 136226511 Ki = 3300 nM T15745 C8ZQ2U 141736359 IC50 = 12160 nM T15745 C5VNM4 141736367 IC50 > 20000 nM T15745 C96NCH 145950955 IC50 > 20000 nM T15745 C3ZV1O 145952497 IC50 > 20000 nM T15745 CTE74G 145954441 IC50 > 20000 nM T15745 CN5YO3 145957310 IC50 > 20000 nM T15745 C7C5WL 145958595 IC50 = 1690 nM T15745 D02KSN 91827353 IC50 = 1070 nM T15745 D03XXT 72201027 IC50 > 20000 nM T15745 D07HET 50967109 IC50 = 26000 nM T15745 D09HBR 135566899 Ki = 3290 nM T15745 D0I4FP 91654625 IC50 = 180 nM T15745 D0T3WL 73010930 IC50 = 430 nM T69612 D06GDY 43815 IC50 > 100000 nM T69612 D0E3TC 44259 IC50 = 73.3 nM T69612 D03BNU 59604787 IC50 > 10000 nM T69612 D00YYO 118888942 IC50 = 5000 nM T69612 D05PTF 118888905 IC50 > 100000 nM T69612 D0U5IW 118888913 IC50 = 88000 nM T69612 D0YD7S 118888923 IC50 = 40000 nM T69612 D0R2TM 5287736 IC50 = 160 nM T69612 D0T3ME 156422 IC50 > 30000 nM T69612 C48HIZ 11155477 IC50 = 2200 nM T69612 CM6DO0 11233873 IC50 > 100000 nM T69612 CQR05P 11494718 IC50 = 5700 nM T69612 CHT93E 11502159 IC50 > 30000 nM T69612 C5VPH9 16129448 IC50 = 4950 nM T69612 CA1D9Q 16155233 IC50 = 1600 nM T69612 CB3Z8Q 25210972 IC50 = 3200 nM T69612 C16ISR 25218571 IC50 = 3200 nM T69612 CP81DI 25218601 IC50 = 2500 nM T69612 CG89VQ 44256165 IC50 = 700 nM T69612 CF8U5T 44256167 IC50 = 660 nM T69612 C0SE3Q 44256203 IC50 = 500 nM T69612 CT2MO1 44256205 IC50 = 1760 nM T69612 CI21MW 44256238 IC50 = 120 nM T69612 CUM54B 44256240 IC50 = 1050 nM T69612 CZ7V6J 44256242 IC50 = 3500 nM T69612 CX9NJ8 44256244 IC50 = 5050 nM T69612 CWK6F0 44256275 IC50 = 3220 nM T69612 CU03ZE 44256279 IC50 = 4300 nM T69612 CE3Y6K 44256281 IC50 = 810 nM T69612 C1QXF2 44256314 IC50 = 3700 nM T69612 C2MS6Q 44256343 IC50 = 4700 nM T69612 C2IJ6R 44256345 IC50 = 1250 nM T69612 CN35VU 44256347 IC50 = 4200 nM T69612 C7NB5X 44256371 IC50 = 520 nM T69612 CV1X8T 44256373 IC50 = 1940 nM T69612 C6UKT1 44256406 IC50 = 6400 nM T69612 CO89LE 44256480 IC50 = 11400 nM T69612 C8NA4L 53384644 IC50 > 30000 nM T69612 C61EBT 60141028 IC50 = 450 nM T69612 CFQ1U4 60142431 IC50 = 3220 nM T69612 C18CIG 60142559 IC50 = 880 nM T69612 C6DHB7 60142693 IC50 = 1660 nM T69612 C1FOD2 60142694 IC50 = 880 nM T69612 CAXK87 60142952 IC50 = 14000 nM T69612 CBCE37 60142954 IC50 = 870 nM T69612 CL0N9F 60143086 IC50 = 2200 nM T69612 CZT65A 60143089 IC50 = 210 nM T69612 C37NKO 67129970 IC50 = 8120 nM T69612 CK80LJ 67130050 IC50 = 9960 nM T69612 CV63UL 67240318 IC50 > 10000 nM T69612 C7GRV2 68755406 IC50 > 10000 nM T69612 CN8F4V 70690082 IC50 = 3100 nM T69612 CR5N7S 72724699 IC50 = 4500 nM T69612 C3R6FU 72724978 IC50 = 3400 nM T69612 C25OTJ 72725039 IC50 = 6900 nM T69612 C3I4GZ 72725092 IC50 = 1140 nM T69612 CFEA16 72725094 IC50 = 1310 nM T69612 CRWU68 72725096 IC50 = 7900 nM T69612 CS7I6A 72725098 IC50 = 5700 nM T69612 C8XK0I 72725161 IC50 = 4000 nM T69612 C3LF8A 72725163 IC50 = 3600 nM T69612 CA6WD3 72725165 IC50 = 1200 nM T69612 C3KWN2 72725221 IC50 = 550 nM T69612 C6L5TE 72725225 IC50 = 3490 nM T69612 C6UFA2 72725284 IC50 = 4200 nM T69612 CN8X5K 72725286 IC50 = 2830 nM T69612 CQH30J 72725289 IC50 = 640 nM T69612 CWUN78 72725404 IC50 = 2090 nM T69612 C78TKB 72725451 IC50 = 5100 nM T69612 C1NI9K 72725453 IC50 = 360 nM T69612 CSY5U6 72725501 IC50 = 2210 nM T69612 CGNJ85 72725616 IC50 = 140 nM T69612 CC47ON 76331813 IC50 = 1780 nM T69612 CF9PB2 77105902 IC50 = 63000 nM T69612 CN8V5D 118875292 IC50 > 100000 nM T69612 CPFQ10 118888903 IC50 > 100000 nM T69612 CU2NO8 118888904 IC50 > 100000 nM T69612 CHXW78 118888907 IC50 = 12000 nM T69612 CPVX20 118888909 IC50 > 100000 nM T69612 CG8IB3 118888910 IC50 = 58000 nM T69612 C7L9DW 118888912 IC50 = 2300 nM T69612 CH4KC3 118888914 IC50 = 2800 nM T69612 CQI01Y 118888915 IC50 > 100000 nM T69612 C6P3LQ 118888916 IC50 > 100000 nM T69612 CNH3X7 118888917 IC50 = 4700 nM T69612 CW7E1Z 118888918 IC50 = 68000 nM T69612 C2XEP7 118888920 IC50 = 1700 nM T69612 CC8U5M 118888921 IC50 = 1800 nM T69612 CX9NT0 118888922 IC50 = 19000 nM T69612 C5T9WU 118888924 IC50 = 13000 nM T69612 CQP67H 118888925 IC50 = 19000 nM T69612 CT2U0M 118888926 IC50 = 66000 nM T69612 CYN50X 118888927 IC50 = 3500 nM T69612 C61BRC 118888929 IC50 = 3800 nM T69612 C7CXF9 118888930 IC50 > 100000 nM T69612 CL57HO 118888931 IC50 = 71000 nM T69612 C60FYM 118888932 IC50 = 19000 nM T69612 CTP32I 118888933 IC50 > 100000 nM T69612 CTC29U 118888934 IC50 = 260 nM T69612 CU6E8W 118888935 IC50 = 44000 nM T69612 C1TQW8 118888936 IC50 > 100000 nM T69612 CWK0V8 118888937 IC50 = 380 nM T69612 C2QE6K 118888938 IC50 > 100000 nM T69612 C15LEY 118888939 IC50 = 6200 nM T69612 CKL47W 118888940 IC50 = 800 nM T69612 CRUI71 118888941 IC50 = 380 nM T69612 CEQ5D3 118888943 IC50 = 8100 nM T69612 CW2QI4 127044088 IC50 > 100000 nM T69612 CR8UX2 127044089 IC50 > 100000 nM T69612 CNV07O 130338701 IC50 > 100000 nM T69612 C3KP5Y 134133467 IC50 = 61300 nM T69612 CY5E0S 134138965 IC50 = 3900 nM T69612 CDG62X 134144831 IC50 = 7400 nM T69612 C0AV2T 134146492 IC50 = 2100 nM T69612 CF8D2L 134153434 IC50 = 9400 nM T69612 C06NOP 136227777 IC50 = 530 nM T69612 CI1E8V 137634241 IC50 > 10000 nM T69612 CG2JO7 137638433 IC50 = 1500 nM T69612 CX5BK1 137647477 IC50 = 21000 nM T69612 C8R0JP 137654554 IC50 > 30000 nM T69612 CFW48S 145967659 IC50 = 38000 nM T69612 CYNP76 145967873 IC50 = 27000 nM T69612 C42CGS 145968147 IC50 = 25000 nM T69612 CGY7E2 145968197 IC50 = 77000 nM T69612 CEM07I 145969035 IC50 = 27000 nM T69612 CUC7I9 145969093 IC50 > 100000 nM T69612 CL1XI2 145969315 IC50 = 18000 nM T69612 CJ3VX0 145969342 IC50 > 100000 nM T69612 C3S6TZ 145969486 IC50 = 16000 nM T69612 CK96OA 145969519 IC50 = 1900 nM T69612 CTD7P8 145969653 IC50 > 100000 nM T69612 CG4KN3 145969683 IC50 = 21000 nM T69612 CEY10F 145970038 IC50 > 100000 nM T69612 CZ96VC 145970244 IC50 > 100000 nM T69612 CM9DW8 145970713 IC50 = 21000 nM T69612 CHM13S 145970814 IC50 > 100000 nM T69612 CL9MI5 145970825 IC50 = 2400 nM T69612 CE39PX 145970840 IC50 = 6300 nM T69612 CI19WX 145970891 IC50 = 9500 nM T69612 CC13LU 145970939 IC50 = 9300 nM T69612 CXQ19A 145971104 IC50 > 100000 nM T69612 CQJ09K 145986806 IC50 = 6100 nM T69612 C6W9SK 145987049 IC50 > 100000 nM T69612 C2MD1Q 155513187 IC50 > 10000 nM T69612 C3C6BJ 155519032 IC50 = 19000 nM T69612 C04ABU 155520084 IC50 > 100000 nM T69612 CLX1C2 155520756 IC50 > 100000 nM T69612 C8ULA4 155520943 IC50 = 5500 nM T69612 CUE34J 155525149 IC50 = 300 nM T69612 CM0N4H 155525309 IC50 = 22000 nM T69612 CX5UJ8 155530668 IC50 = 220 nM T69612 C3SV1L 155537345 IC50 = 220 nM T69612 CV04YS 155541038 IC50 = 17000 nM T69612 C8VP2Y 155548752 IC50 > 100000 nM T69612 C90GHF 155552339 IC50 = 5900 nM T69612 C3AVC1 155553988 IC50 = 4800 nM T69612 C96ZTB 155556754 IC50 = 1100 nM T69612 C7IT2V 155560286 IC50 > 100000 nM T69612 C3U1NE 155564829 IC50 = 78000 nM T69612 CJ23NM 155568844 IC50 = 7100 nM T69612 D04CUA 44256277 IC50 = 59 nM T69612 D0U8UK 11677079 IC50 = 2300 nM T47101 D01PZD 5329098 IC50 = 4200 nM T47101 D03ZBT 11626560 IC50 > 1000 nM T47101 D09GDD 11167602 IC50 = 1.5 nM T47101 D0B0AX 5328127 IC50 = 48 nM T47101 D0C4RB 36314 IC50 > 10000 nM T47101 D0E6XR 3062316 IC50 = 880 nM T47101 D0G6QF 3081361 IC50 = 2310 nM T47101 D0H0EQ 24826799 IC50 = 0.7 nM T47101 D0IQ6P 25102847 IC50 = 11.3 nM T47101 D0J9ZR 4477 IC50 = 13100 nM T47101 D0R0MW 5329102 IC50 = 170 nM T47101 D0W5HK 216239 IC50 = 670 nM T47101 D00DRL 44137946 IC50 = 65 nM T47101 D00UZR 5330286 IC50 > 10000 nM T47101 D02RJY 11442891 IC50 = 47 nM T47101 D02UFQ 11620908 IC50 > 10000 nM T47101 D02WVT 25031915 IC50 = 17.5 nM T47101 D03HUX 49792852 IC50 > 10000 nM T47101 D03LWG 53235510 IC50 = 0.59 nM T47101 D05PZB 135398495 IC50 = 10 nM T47101 D07EHV 44814409 IC50 > 10000 nM T47101 D07HPJ 11476171 IC50 = 4300 nM T47101 D07PNT 10433653 IC50 = 4 nM T47101 D08EQD 118036971 IC50 > 10000 nM T47101 D08HOM 46207586 IC50 = 188 nM T47101 D0A1AQ 5329099 IC50 = 1950 nM T47101 D0D4VV 46944259 IC50 = 0.3 nM T47101 D0D6XT 118029202 IC50 = 320 nM T47101 D0E3TC 44259 IC50 = 3.89 nM T47101 D0FD6D 11751922 IC50 = 13 nM T47101 D0H9FR 118295624 IC50 = 0.6 nM T47101 D0HS5V 11234052 IC50 = 148 nM T47101 D0IQ0Z 46885626 IC50 = 76 nM T47101 D0M0XB 10302451 IC50 > 10000 nM T47101 D0M9QZ 11485656 IC50 = 5479 nM T47101 D0NW0T 67462786 IC50 = 1.2 nM T47101 D0O0LS 25141092 IC50 > 1000 nM T47101 D0P1CV 46191454 IC50 > 10000 nM T47101 D0Q9UX 16718576 IC50 = 1207 nM T47101 D0S7HM 16041424 IC50 = 93 nM T47101 D0VF6E 1401 IC50 = 19 nM T47101 D0XT0W 66555680 IC50 = 9.3 nM T47101 D03BNU 59604787 IC50 > 10000 nM T47101 D0LF0O 135441202 IC50 < 5000 nM T47101 D0YK9D 9956119 IC50 > 5000 nM T47101 D0H4GI 10275001 IC50 = 162 nM T47101 D0H8KG 5311382 IC50 = 43 nM T47101 D0L5YF 5329032 IC50 > 100000 nM T47101 D0T3ME 156422 IC50 = 15000 nM T47101 C0ISD9 12855 IC50 > 50000 nM T47101 COI41C 84657 IC50 > 50000 nM T47101 CPLW61 136693 IC50 > 50000 nM T47101 C6Y9CV 151193 IC50 > 10000 nM T47101 CZ18BP 182029 IC50 > 50000 nM T47101 CY1UK0 304268 IC50 > 50000 nM T47101 CK0L4O 442514 IC50 = 320 nM T47101 C4MNG8 445840 IC50 = 6700 nM T47101 C1ZG2U 449087 IC50 > 10000 nM T47101 C78IXN 563347 IC50 > 50000 nM T47101 C9LG4T 639427 IC50 > 50000 nM T47101 C75EDQ 644355 IC50 > 10000 nM T47101 C5HPF3 644356 IC50 > 10000 nM T47101 CE1US5 652633 IC50 > 50000 nM T47101 C2NE1O 703493 IC50 > 50000 nM T47101 C2S9PG 703747 IC50 = 6300 nM T47101 CQRW97 703930 IC50 = 4300 nM T47101 CVZ6D8 705189 IC50 = 4300 nM T47101 C98PSQ 705972 IC50 = 18200 nM T47101 C9HY2V 709070 IC50 > 30000 nM T47101 CH7R8E 709073 IC50 > 30000 nM T47101 CX54PC 709076 IC50 = 5000 nM T47101 CU21GT 709079 IC50 > 30000 nM T47101 CD1U3R 709202 IC50 = 3000 nM T47101 CET1C2 710688 IC50 > 50000 nM T47101 CKZT51 724946 IC50 = 2500 nM T47101 CLJ5X1 725352 IC50 = 1660 nM T47101 CRJT26 733564 IC50 = 700 nM T47101 CS1M4H 733565 IC50 = 180 nM T47101 CKU8S5 733567 IC50 = 1200 nM T47101 CSK73A 733568 IC50 = 160 nM T47101 C38YBV 733570 IC50 = 500 nM T47101 CNG26L 733958 IC50 > 30000 nM T47101 CO42IV 737733 IC50 > 50000 nM T47101 CK2E5S 739094 IC50 > 50000 nM T47101 C3XKO9 743942 IC50 > 50000 nM T47101 CG6O9V 794657 IC50 > 50000 nM T47101 CXDO32 852492 IC50 > 50000 nM T47101 C8WJR7 965312 IC50 = 36000 nM T47101 CQT71Y 1179824 IC50 > 30000 nM T47101 CB0C5A 1188994 IC50 > 30000 nM T47101 C1ORJ6 1189380 IC50 > 30000 nM T47101 C72TVI 1189381 IC50 = 11000 nM T47101 C7RD4S 1191830 IC50 = 3000 nM T47101 COX7Y1 1191831 IC50 = 500 nM T47101 C37MEI 1193936 IC50 = 12500 nM T47101 COB86I 1474850 IC50 = 58000 nM T47101 C2GSN6 1475052 IC50 > 100000 nM T47101 CQ6TW7 1540283 IC50 > 50000 nM T47101 CLI56S 1567987 IC50 > 30000 nM T47101 C7WPA5 1586853 IC50 = 1600 nM T47101 CQG37S 1645520 IC50 = 1250 nM T47101 CAV19R 2360773 IC50 > 10000 nM T47101 C85KVI 2771646 IC50 > 50000 nM T47101 C8SDU2 2773197 IC50 > 50000 nM T47101 CRP7B3 2788649 IC50 = 3200 nM T47101 CT7W4M 2927432 IC50 = 50000 nM T47101 CHC5I0 2971839 IC50 > 10000 nM T47101 CFY1D0 2974957 IC50 > 10000 nM T47101 C2B6VQ 3693861 IC50 > 30000 nM T47101 CXCP46 4327052 IC50 > 50000 nM T47101 CB3G6R 4913175 IC50 = 8000 nM T47101 CQVC06 4962150 IC50 > 50000 nM T47101 CA9E8N 4962189 IC50 > 50000 nM T47101 CMC76E 5327864 IC50 = 1300 nM T47101 CP94NE 5327865 IC50 = 5800 nM T47101 C43JFT 5327866 IC50 > 50000 nM T47101 C5D2VK 5327867 IC50 > 50000 nM T47101 C4ZW0Q 5327868 IC50 = 2500 nM T47101 CY82TU 5327869 IC50 = 960 nM T47101 CL4OG5 5327870 IC50 = 700 nM T47101 CYGA64 5327871 IC50 = 4480 nM T47101 CZE87D 5327872 IC50 = 6800 nM T47101 C7XOK5 5327873 IC50 = 1660 nM T47101 CQK5Z0 5327874 IC50 = 14000 nM T47101 CS0Q4N 5327875 IC50 > 50000 nM T47101 CI96EG 5327876 IC50 = 13900 nM T47101 CT86OE 5327877 IC50 = 1400 nM T47101 C23EZX 5327878 IC50 = 380 nM T47101 C63SAG 5327879 IC50 = 320 nM T47101 CT94BD 5327880 IC50 = 240 nM T47101 CNRS28 5327881 IC50 = 3210 nM T47101 CD43FT 5327882 IC50 = 3150 nM T47101 CX39AM 5327883 IC50 = 6530 nM T47101 CZWG61 5327884 IC50 = 580 nM T47101 C3P8CG 5327885 IC50 = 30 nM T47101 CWZ8H3 5327886 IC50 = 210 nM T47101 CC7VR3 5327887 IC50 = 150 nM T47101 CG7Q3R 5327888 IC50 = 540 nM T47101 CYRW80 5327889 IC50 = 190 nM T47101 C7W8IJ 5327890 IC50 = 110 nM T47101 CJ28SO 5327891 IC50 = 3000 nM T47101 C82PDN 5327892 IC50 = 2400 nM T47101 C52MYD 5327893 IC50 = 910 nM T47101 C4ET5H 5327894 IC50 = 3200 nM T47101 CJ5VO8 5327895 IC50 = 370 nM T47101 CDA78E 5327896 IC50 = 410 nM T47101 CQ0ZP3 5327897 IC50 = 180 nM T47101 C7KIT4 5327898 IC50 = 150 nM T47101 COQH79 5327899 IC50 = 450 nM T47101 C9R8DP 5327900 IC50 = 430 nM T47101 CJCE40 5327901 IC50 = 1500 nM T47101 CVB9L3 5327902 IC50 = 33600 nM T47101 C7EK0Z 5327903 IC50 = 2600 nM T47101 C4ZD2M 5327904 IC50 = 55 nM T47101 CK58VC 5327905 IC50 = 66 nM T47101 C85BRY 5327906 IC50 = 34 nM T47101 CVDS17 5327907 IC50 = 33 nM T47101 CLH9Y3 5327908 IC50 = 30 nM T47101 C04BUF 5327909 IC50 = 30 nM T47101 CT7RL1 5327910 IC50 = 40 nM T47101 CBJV81 5327912 IC50 = 46 nM T47101 CDO81N 5327913 IC50 = 39 nM T47101 CA7U3O 5327914 IC50 = 28 nM T47101 CT91PJ 5327915 IC50 = 49 nM T47101 CN71AK 5327916 IC50 = 110 nM T47101 C5JI1A 5327917 IC50 = 61 nM T47101 C4CWI1 5327918 IC50 = 110 nM T47101 CPT61U 5328112 IC50 = 110 nM T47101 CMW3F8 5328113 IC50 = 3000 nM T47101 CBZ97E 5328114 IC50 = 2400 nM T47101 CXR9K1 5328115 IC50 = 82 nM T47101 CT3N1W 5328116 IC50 = 13000 nM T47101 CM0H5O 5328117 IC50 = 400 nM T47101 CW1Q8K 5328118 IC50 = 18000 nM T47101 CHO9N3 5328119 IC50 = 340 nM T47101 C17QCT 5328120 IC50 = 13000 nM T47101 C7UJH5 5328121 IC50 = 290 nM T47101 CN4Y5V 5328122 IC50 = 8300 nM T47101 CCI13D 5328123 IC50 = 190 nM T47101 C8LGY6 5328124 IC50 > 50000 nM T47101 CDM98R 5328125 IC50 = 710 nM T47101 CDH5C1 5328126 IC50 = 230 nM T47101 CI7VF4 5328129 IC50 = 1300 nM T47101 CP4K1A 5328130 IC50 = 1800 nM T47101 CEGO42 5328131 IC50 = 130 nM T47101 CNT01S 5328132 IC50 = 77 nM T47101 CDY2O3 5328134 IC50 = 49 nM T47101 CC1O0M 5328135 IC50 = 48 nM T47101 CZ95IT 5328136 IC50 = 43 nM T47101 C14LVT 5328137 IC50 = 110 nM T47101 C6WC2I 5328139 IC50 = 75 nM T47101 C9PBI3 5328141 IC50 = 2000 nM T47101 C8TEQ0 5328143 IC50 = 210 nM T47101 CC1KQ8 5328145 IC50 = 72 nM T47101 C4K7JS 5328147 IC50 = 60 nM T47101 CKB92Q 5328148 IC50 = 450 nM T47101 COT45A 5328149 IC50 = 51 nM T47101 C7POG3 5328151 IC50 = 35 nM T47101 C1QTZ0 5328152 IC50 = 140 nM T47101 CJR6K4 5328153 IC50 = 53 nM T47101 C9ZGN8 5328154 IC50 = 35 nM T47101 CM9ZO8 5328155 IC50 = 34 nM T47101 CB5P9H 5328156 IC50 = 420 nM T47101 CF3AM9 5328157 IC50 = 62 nM T47101 CT9SO8 5328158 IC50 = 29 nM T47101 C6G7YD 5328159 IC50 = 120 nM T47101 C7QH2V 5328160 IC50 = 67 nM T47101 CB0D7I 5328161 IC50 = 75 nM T47101 CYA9N6 5328162 IC50 = 5500 nM T47101 C5EN6O 5328163 IC50 = 84 nM T47101 COL3B8 5328164 IC50 = 120 nM T47101 CCQA46 5328165 IC50 = 110 nM T47101 CU7TM3 5328166 IC50 = 610 nM T47101 CIL71E 5328167 IC50 = 600 nM T47101 CM2BH6 5328168 IC50 = 110 nM T47101 CZD03I 5328169 IC50 = 67 nM T47101 CMZ40L 5328170 IC50 = 63 nM T47101 CJA36I 5328171 IC50 = 74 nM T47101 CQ9LH6 5328172 IC50 = 300 nM T47101 C1M9NK 5328173 IC50 = 27000 nM T47101 C1HGR7 5328175 IC50 = 260 nM T47101 CIT23N 5328176 IC50 = 2700 nM T47101 C0TDG9 5328177 IC50 = 130 nM T47101 CB2U0H 5328178 IC50 = 3700 nM T47101 C1X8RH 5328179 IC50 = 8000 nM T47101 C6EHD0 5328180 IC50 = 6800 nM T47101 CE64IZ 5328181 IC50 = 68 nM T47101 CE64YI 5328183 IC50 = 2500 nM T47101 C0C4UO 5328184 IC50 = 100 nM T47101 C0DYW6 5328185 IC50 = 320 nM T47101 CURM29 5328426 IC50 > 50000 nM T47101 CR8BD9 5328427 IC50 > 50000 nM T47101 C95XHY 5328428 IC50 > 50000 nM T47101 CI9SD6 5328429 IC50 > 50000 nM T47101 C2YF6I 5328430 IC50 > 50000 nM T47101 C4RPU3 5328431 IC50 > 50000 nM T47101 C1V3KD 5328432 IC50 > 50000 nM T47101 C90WGE 5328433 IC50 > 50000 nM T47101 CB04XV 5328434 IC50 > 50000 nM T47101 C6RCA0 5328435 IC50 > 50000 nM T47101 CDBZ89 5328436 IC50 > 50000 nM T47101 CJ93IF 5328437 IC50 = 50000 nM T47101 CK6FN0 5328438 IC50 = 50000 nM T47101 CU84KM 5328439 IC50 = 50000 nM T47101 C75HYE 5328440 IC50 > 50000 nM T47101 COV4H3 5328441 IC50 > 50000 nM T47101 CIXO42 5328442 IC50 > 50000 nM T47101 CLI01G 5328443 IC50 = 35000 nM T47101 CQY5R1 5328444 IC50 > 50000 nM T47101 CA13OP 5328445 IC50 > 50000 nM T47101 CE2LM5 5328446 IC50 = 50000 nM T47101 CZ29RL 5328447 IC50 > 50000 nM T47101 CMZL20 5328448 IC50 > 50000 nM T47101 C8BF4V 5328449 IC50 = 5800 nM T47101 CO9B0X 5328450 IC50 > 50000 nM T47101 CYK1J0 5328451 IC50 = 50000 nM T47101 CLM85U 5328452 IC50 > 50000 nM T47101 CUK80H 5328454 IC50 > 50000 nM T47101 CW7PL6 5328455 IC50 > 50000 nM T47101 CVH4A8 5328456 IC50 > 50000 nM T47101 C90UTH 5328457 IC50 > 50000 nM T47101 C0Z8KJ 5328458 IC50 > 50000 nM T47101 CK5C6R 5328459 IC50 > 50000 nM T47101 CF28VK 5328460 IC50 > 50000 nM T47101 C4TFU0 5328461 IC50 > 50000 nM T47101 CB0CQ7 5328462 IC50 > 50000 nM T47101 CZSF67 5328463 IC50 > 50000 nM T47101 C18XOD 5328464 IC50 > 50000 nM T47101 C0TNX7 5328465 IC50 = 50000 nM T47101 C3AU7X 5328467 IC50 = 51000 nM T47101 CLC10K 5328468 IC50 = 28000 nM T47101 C10RHA 5328469 IC50 = 6600 nM T47101 C39HSR 5328470 IC50 = 10000 nM T47101 CXP7C0 5328471 IC50 = 14000 nM T47101 C1TW8P 5328472 IC50 > 50000 nM T47101 C2WC7J 5328473 IC50 = 49000 nM T47101 CN74WU 5328474 IC50 > 50000 nM T47101 C6VYE2 5328475 IC50 > 50000 nM T47101 C3L6KP 5328476 IC50 > 50000 nM T47101 CA3N2Z 5328477 IC50 = 50000 nM T47101 C7RP2V 5328478 IC50 > 50000 nM T47101 C5O7NC 5328479 IC50 > 50000 nM T47101 C0MES9 5328480 IC50 = 39000 nM T47101 CQ8PF0 5328481 IC50 > 50000 nM T47101 C9ELG0 5328482 IC50 > 50000 nM T47101 C2FZP9 5328483 IC50 = 50000 nM T47101 CIV4K8 5328484 IC50 = 50000 nM T47101 C6FBN7 5328485 IC50 > 50000 nM T47101 CNA3Y7 5328486 IC50 > 50000 nM T47101 CC9ON2 5328487 IC50 > 50000 nM T47101 CE6YD0 5328488 IC50 > 50000 nM T47101 C7V2YB 5328489 IC50 = 40000 nM T47101 CDF4P8 5328490 IC50 > 50000 nM T47101 C8INH7 5328491 IC50 > 50000 nM T47101 C2PEV1 5328492 IC50 = 5300 nM T47101 CKR29P 5328493 IC50 = 6500 nM T47101 CLZT78 5328497 IC50 > 50000 nM T47101 C8C0RL 5328498 IC50 = 35000 nM T47101 CGW0I4 5328499 IC50 = 50000 nM T47101 CO4W7V 5328500 IC50 = 50000 nM T47101 CI5E6B 5328501 IC50 = 35000 nM T47101 CB3J1O 5328502 IC50 = 25000 nM T47101 CH2F1N 5328503 IC50 = 18000 nM T47101 C4AUK6 5328504 IC50 = 15000 nM T47101 CFSN21 5328505 IC50 = 27000 nM T47101 CWQO83 5328506 IC50 = 45000 nM T47101 CG5M7U 5328507 IC50 = 4100 nM T47101 C4FE0B 5328508 IC50 = 6800 nM T47101 CJM61R 5328509 IC50 = 28000 nM T47101 CIY48D 5328510 IC50 = 9800 nM T47101 CM3D5O 5328511 IC50 = 12000 nM T47101 CN8IE6 5328513 IC50 > 50000 nM T47101 C1XMV2 5328514 IC50 = 27000 nM T47101 CKEY79 5328515 IC50 = 24000 nM T47101 CT65IH 5328516 IC50 > 50000 nM T47101 CA18OW 5328517 IC50 = 1900 nM T47101 CJX18A 5328518 IC50 > 50000 nM T47101 CI1BS6 5328519 IC50 > 50000 nM T47101 C2W7DN 5328520 IC50 > 50000 nM T47101 CDL94I 5328521 IC50 > 50000 nM T47101 CO04IH 5328522 IC50 > 50000 nM T47101 C7HPN8 5328523 IC50 > 50000 nM T47101 CPZD13 5328524 IC50 > 50000 nM T47101 C1M2CY 5328525 IC50 = 25000 nM T47101 CS3CR5 5328526 IC50 = 11000 nM T47101 CM9EJ7 5328527 IC50 = 27000 nM T47101 CJE94R 5328528 IC50 > 50000 nM T47101 C2NE5X 5328529 IC50 > 50000 nM T47101 CXR8Z6 5328530 IC50 > 50000 nM T47101 CQH57F 5328531 IC50 = 22000 nM T47101 C0MW1I 5328532 IC50 = 50000 nM T47101 CFWZ98 5328533 IC50 = 11000 nM T47101 CK4L8D 5328534 IC50 = 25000 nM T47101 C0TX2I 5328592 IC50 = 4500 nM T47101 CUE30V 5328700 IC50 = 380 nM T47101 C9IH8T 5328701 IC50 = 210 nM T47101 CL61RQ 5328702 IC50 > 50000 nM T47101 C9T8GP 5328703 IC50 = 33000 nM T47101 CI9B1T 5328704 IC50 = 150 nM T47101 C8VEP0 5328705 IC50 = 80 nM T47101 C4QZ1J 5328706 IC50 = 80 nM T47101 CR0UB3 5328707 IC50 = 170 nM T47101 C4GCM3 5328708 IC50 = 170 nM T47101 CFG6I9 5328709 IC50 = 110 nM T47101 CY12MK 5328710 IC50 = 570 nM T47101 C13KGU 5328711 IC50 = 230 nM T47101 C7XN8T 5328712 IC50 = 210 nM T47101 CFK34R 5328713 IC50 = 2200 nM T47101 C37VOE 5328714 IC50 = 3500 nM T47101 CBH91D 5328715 IC50 = 2200 nM T47101 COL47I 5328716 IC50 = 130 nM T47101 COI8H6 5328717 IC50 = 250 nM T47101 C8UK0W 5328718 IC50 = 210 nM T47101 CO1EU7 5328719 IC50 = 120 nM T47101 CX9D7E 5328720 IC50 = 42 nM T47101 CR4VJ8 5328721 IC50 = 8700 nM T47101 CTV12Y 5328722 IC50 = 1900 nM T47101 C50CGB 5328723 IC50 = 170 nM T47101 CEW4B8 5328724 IC50 = 72 nM T47101 CCKV98 5328725 IC50 = 440 nM T47101 CN9ST1 5328726 IC50 > 50000 nM T47101 CDZF47 5328727 IC50 > 50000 nM T47101 CZN6F4 5328728 IC50 > 50000 nM T47101 CKD93O 5328729 IC50 > 50000 nM T47101 C5ICG9 5328730 IC50 > 50000 nM T47101 CM25VZ 5328731 IC50 > 50000 nM T47101 C56SHL 5328732 IC50 > 50000 nM T47101 CPL1U9 5328734 IC50 = 180 nM T47101 C5R9DV 5328990 IC50 = 17000 nM T47101 CDNP54 5328991 IC50 = 1300 nM T47101 C6J5YD 5328992 IC50 = 1900 nM T47101 CY5L7F 5328993 IC50 = 2800 nM T47101 CCV0B4 5328994 IC50 = 150 nM T47101 C3A1ER 5328995 IC50 = 120 nM T47101 CA05KW 5328996 IC50 = 200 nM T47101 CF0PG3 5328997 IC50 = 95 nM T47101 C68UKW 5328998 IC50 = 29 nM T47101 CU4XT5 5328999 IC50 = 42 nM T47101 CPK58V 5329000 IC50 = 510 nM T47101 C10WHP 5329001 IC50 = 25 nM T47101 C7HB6C 5329002 IC50 = 61 nM T47101 C5D4WA 5329003 IC50 = 160 nM T47101 CWX63A 5329004 IC50 = 31 nM T47101 CQL3C9 5329005 IC50 > 100000 nM T47101 CFW19M 5329009 IC50 > 100000 nM T47101 C2FO4B 5329010 IC50 = 2500 nM T47101 CZU0K3 5329011 IC50 = 27000 nM T47101 C21WXV 5329012 IC50 = 7000 nM T47101 CJ68OQ 5329013 IC50 = 7400 nM T47101 CEJR83 5329014 IC50 > 100000 nM T47101 COS5M9 5329015 IC50 = 16000 nM T47101 CKFS07 5329016 IC50 = 1400 nM T47101 CC1EO4 5329017 IC50 = 9300 nM T47101 CGC01T 5329018 IC50 = 9400 nM T47101 C1XJL0 5329019 IC50 = 19000 nM T47101 C9SZ4Q 5329020 IC50 = 6700 nM T47101 C5DO1Y 5329021 IC50 = 1500 nM T47101 C2YDI8 5329022 IC50 = 20000 nM T47101 CW3OV5 5329023 IC50 > 50000 nM T47101 C6HSX8 5329024 IC50 > 33000 nM T47101 CP37NS 5329025 IC50 = 2600 nM T47101 C3VHF6 5329026 IC50 = 1600 nM T47101 CSRF48 5329027 IC50 = 25000 nM T47101 CB6V5Y 5329028 IC50 = 1800 nM T47101 C6AN1O 5329029 IC50 > 50000 nM T47101 C04EAP 5329030 IC50 = 40000 nM T47101 C1Y5QP 5329031 IC50 > 100000 nM T47101 C4VLR8 5329033 IC50 = 6100 nM T47101 CLT7J9 5329034 IC50 = 45000 nM T47101 C9VX8C 5329040 IC50 = 19000 nM T47101 CK6T4U 5329042 IC50 = 13500 nM T47101 CA81XO 5329045 IC50 = 1700 nM T47101 C4T3MO 5329046 IC50 = 1500 nM T47101 CQ15KR 5329049 IC50 = 12300 nM T47101 C49KNS 5329050 IC50 = 2500 nM T47101 C3C1EZ 5329051 IC50 = 1900 nM T47101 C0H5XL 5329052 IC50 = 4100 nM T47101 CW0KA8 5329053 IC50 = 2100 nM T47101 COEN93 5329054 IC50 = 2700 nM T47101 CATX52 5329055 IC50 = 1800 nM T47101 CEQP41 5329056 IC50 = 1800 nM T47101 CDV4C9 5329057 IC50 = 5000 nM T47101 C9I7WT 5329100 IC50 = 4200 nM T47101 CMWB28 5329101 IC50 = 880 nM T47101 CGX50J 5329104 IC50 = 730 nM T47101 C2VX0H 5329105 IC50 = 1600 nM T47101 CK71MQ 5329106 IC50 = 3900 nM T47101 CL0Q4S 5329107 IC50 = 200 nM T47101 C6YRH8 5329108 IC50 = 2600 nM T47101 CFP59Y 5329109 IC50 = 3100 nM T47101 CSY10K 5329111 IC50 = 3700 nM T47101 CV7FG2 5329112 IC50 = 160 nM T47101 C4VQ2R 5329113 IC50 = 110 nM T47101 C2SQL0 5329114 IC50 = 180 nM T47101 CNI13Q 5329115 IC50 = 110 nM T47101 C1JF3N 5329116 IC50 = 1100 nM T47101 C19GHD 5329117 IC50 > 50000 nM T47101 C6C8RV 5329118 IC50 = 1400 nM T47101 C5V8FR 5329119 IC50 = 1670 nM T47101 CYU89T 5329120 IC50 = 340 nM T47101 CDU9H6 5329121 IC50 = 1130 nM T47101 CMAV05 5329122 IC50 = 270 nM T47101 CG8B3E 5329123 IC50 = 1620 nM T47101 CW5U4J 5329124 IC50 = 890 nM T47101 C39FIH 5329125 IC50 = 11220 nM T47101 CMY9D6 5329126 IC50 = 7760 nM T47101 C6VO5Z 5329127 IC50 = 11220 nM T47101 CM7B2T 5329128 IC50 = 360 nM T47101 C9GXO6 5329129 IC50 = 3970 nM T47101 CP5AI7 5329130 IC50 = 20250 nM T47101 C4I3ZO 5329131 IC50 = 670 nM T47101 C8IF1G 5329132 IC50 = 1650 nM T47101 CE68LC 5329133 IC50 = 16000 nM T47101 C0JW3Y 5329134 IC50 = 30 nM T47101 CO7J2A 5329135 IC50 = 80 nM T47101 CQ4TP5 5329136 IC50 = 140 nM T47101 CXQC42 5329137 IC50 = 270 nM T47101 CT94JS 5329138 IC50 = 3680 nM T47101 CNH06M 5329139 IC50 = 770 nM T47101 CRY4Z2 5329140 IC50 = 460 nM T47101 CAPE50 5329141 IC50 = 31600 nM T47101 CFU58A 5329142 IC50 = 1000 nM T47101 C5Q8XK 5329143 IC50 = 130 nM T47101 C8PX4D 5329144 IC50 = 40 nM T47101 C6USQ5 5329145 IC50 = 1600 nM T47101 C56LWT 5329146 IC50 = 2050 nM T47101 CZ16MN 5329147 IC50 = 280 nM T47101 CAN16I 5329148 IC50 = 280 nM T47101 CG4NC2 5329149 IC50 = 25100 nM T47101 CIW70H 5329150 IC50 = 2290 nM T47101 C5FT6A 5329151 IC50 = 1500 nM T47101 CB0N4L 5329152 IC50 = 4000 nM T47101 COFP24 5329153 IC50 = 5760 nM T47101 CGWD98 5329154 IC50 = 10500 nM T47101 C4PD0K 5329156 IC50 = 220 nM T47101 C0RWT8 5329157 IC50 = 310 nM T47101 C3MU5S 5329158 IC50 > 20000 nM T47101 CN6O4R 5329159 IC50 > 20000 nM T47101 CG68DI 5329160 IC50 = 17500 nM T47101 CYR7V0 5329161 IC50 = 17700 nM T47101 C9BXE2 5329162 IC50 > 20000 nM T47101 CY4V5Z 5329163 IC50 = 270 nM T47101 CI64YA 5329164 IC50 = 270 nM T47101 C2ZV0O 5329165 IC50 = 200 nM T47101 CAB53L 5329166 IC50 = 220 nM T47101 CTW9R8 5329167 IC50 = 1080 nM T47101 C8A3TJ 5329168 IC50 = 1270 nM T47101 CVTD82 5329169 IC50 = 1350 nM T47101 CQ5WK1 5329170 IC50 = 80 nM T47101 CNC9T7 5329171 IC50 = 880 nM T47101 CBS40G 5330125 IC50 = 44 nM T47101 CNWK81 5330126 IC50 = 21 nM T47101 CV7GX5 5330127 IC50 = 24 nM T47101 CWAR90 5330128 IC50 = 8 nM T47101 CDG3Z1 5330129 IC50 = 7 nM T47101 C09VSN 5330130 IC50 = 24 nM T47101 CNMJ73 5330131 IC50 = 46 nM T47101 CV4U8Y 5330132 IC50 = 24 nM T47101 C6D7WJ 5330133 IC50 = 6 nM T47101 C2UX4V 5330134 IC50 = 33 nM T47101 CH38FW 5330135 IC50 = 10 nM T47101 CWQ47D 5330136 IC50 = 6 nM T47101 CP2UB6 5330137 IC50 = 2200 nM T47101 CJYX18 5330138 IC50 = 140 nM T47101 CR73WA 5330139 IC50 = 12000 nM T47101 C54VLJ 5330140 IC50 = 7300 nM T47101 C9QO0W 5330141 IC50 = 200 nM T47101 CLD7I9 5330142 IC50 = 120 nM T47101 CZ8G1N 5330143 IC50 = 16 nM T47101 C7K5PV 5330144 IC50 = 26 nM T47101 CK5CG4 5330145 IC50 = 630 nM T47101 CPA63S 5330146 IC50 = 16 nM T47101 CY08DW 5330147 IC50 = 25 nM T47101 C6FAS9 5330148 IC50 = 330 nM T47101 CCGA06 5330149 IC50 = 2400 nM T47101 C9USJ0 5330150 IC50 = 3300 nM T47101 CQX0A3 5330151 IC50 = 1400 nM T47101 CBD8N6 5330152 IC50 = 8400 nM T47101 CX2FO6 5330153 IC50 = 7500 nM T47101 CLI47K 5330157 IC50 = 4 nM T47101 CNI15R 5330158 IC50 = 8 nM T47101 C4IA7N 5330159 IC50 = 10 nM T47101 CSL02W 5330160 IC50 = 9000 nM T47101 CNA8R7 5330161 IC50 = 1100 nM T47101 CF4JU8 5330162 IC50 = 20000 nM T47101 CDY0R5 5330163 IC50 = 7900 nM T47101 CR0GX9 5330164 IC50 = 8700 nM T47101 C37DGR 5330165 IC50 = 7700 nM T47101 CW8G9J 5330166 IC50 = 18 nM T47101 C7Z2YH 5330167 IC50 = 11 nM T47101 CEX9A7 5330168 IC50 = 35 nM T47101 C3I6KF 5330169 IC50 = 38 nM T47101 C5RK3H 5330188 IC50 > 100000 nM T47101 CD7U5B 5330196 IC50 > 100000 nM T47101 CB23PA 5330197 IC50 > 100000 nM T47101 C9NBG7 5330546 IC50 = 200 nM T47101 CM47KI 5351344 IC50 > 10000 nM T47101 CDK3J0 5703619 IC50 = 12 nM T47101 CB7WK3 5938113 IC50 = 9000 nM T47101 CXC62N 6326404 IC50 = 10000 nM T47101 CE60XJ 6326405 IC50 = 2800 nM T47101 CV2KQ1 6326407 IC50 > 33000 nM T47101 CF46XV 6326408 IC50 = 14000 nM T47101 CN2W1U 6488846 IC50 = 5600 nM T47101 CI80BK 9803350 IC50 = 400 nM T47101 CXA5C8 9893493 IC50 = 58 nM T47101 CHB0D2 9982235 IC50 = 18 nM T47101 C7Q5CN 10015651 IC50 = 5100 nM T47101 C7YD1X 10048045 IC50 > 25000 nM T47101 CUJR40 10062694 EC50 = 80 nM T47101 C1JUF8 10073832 IC50 = 100 nM T47101 CIV15Q 10113978 IC50 = 140 nM T47101 C6DC8Q 10275163 IC50 = 700 nM T47101 C8RD3V 10301884 IC50 = 37000 nM T47101 C5CBF9 10320381 IC50 = 70 nM T47101 C07XHY 10388612 IC50 = 20 nM T47101 CQ6OF5 10388672 IC50 = 140 nM T47101 C7HBP6 10429593 IC50 > 10000 nM T47101 C2VPT6 10436729 IC50 = 16 nM T47101 C7PLI5 10478569 IC50 = 19 nM T47101 CJ5M1D 10482445 IC50 = 200 nM T47101 CJO8Q1 10738332 IC50 = 130 nM T47101 COMB49 11155938 IC50 = 27 nM T47101 C7V8JR 11167666 IC50 = 149 nM T47101 CBOP58 11293798 Ki > 10000 nM T47101 CC8J3N 11328182 IC50 = 50 nM T47101 CA6F4L 11352215 IC50 = 33 nM T47101 C26BZX 11362471 Ki > 10000 nM T47101 CG57WD 11374515 IC50 = 28 nM T47101 CWXB93 11397177 Ki > 10000 nM T47101 CQD35C 11419379 IC50 = 110 nM T47101 C7AI2V 11432911 IC50 = 220 nM T47101 C45WKC 11442803 IC50 = 39 nM T47101 CZ9O1A 11455031 IC50 = 68 nM T47101 CJUF06 11464544 IC50 = 160 nM T47101 CTG3D9 11465545 IC50 = 14 nM T47101 C6M9NC 11477626 IC50 = 46 nM T47101 CE39WZ 11488852 IC50 = 84 nM T47101 CACS26 11561968 Ki > 2000 nM T47101 CZ1H0X 11569258 IC50 = 7100 nM T47101 CSM62L 11626920 IC50 = 13000 nM T47101 CK34LS 11632737 IC50 > 5000 nM T47101 CCX2F5 11682611 IC50 = 3 nM T47101 CU0E8O 11690457 Ki > 2000 nM T47101 CU6D3X 11703421 IC50 = 22 nM T47101 CZY05V 11719421 IC50 = 960 nM T47101 CS36BH 11843159 IC50 = 110 nM T47101 C9JT4S 11847343 IC50 = 14 nM T47101 CP2HR6 11948697 IC50 = 10 nM T47101 C60NJV 11948698 IC50 = 47 nM T47101 CY4R6F 11990802 IC50 > 10000 nM T47101 CZHQ54 12988783 IC50 = 10 nM T47101 CN14SK 12988792 IC50 = 30 nM T47101 CXRK13 12988793 IC50 = 4 nM T47101 CV4EZ6 15949611 IC50 > 10000 nM T47101 C7LB4I 15949613 IC50 > 10000 nM T47101 C9TU1O 16046126 IC50 > 1000 nM T47101 C5VPH9 16129448 IC50 = 4060 nM T47101 C0H8UN 16730109 IC50 > 50000 nM T47101 C3YCJ7 16876232 IC50 > 30000 nM T47101 CBKZ97 16876234 IC50 = 5000 nM T47101 CFN6G4 21701597 IC50 = 2100 nM T47101 CF6LA9 22478260 IC50 = 2100 nM T47101 CMRO51 22478297 IC50 = 1900 nM T47101 CBI80A 22664657 IC50 = 51 nM T47101 CP02XA 22664735 IC50 = 10 nM T47101 COB60M 23133320 IC50 = 4300 nM T47101 C9QLP0 23133323 IC50 = 3600 nM T47101 CG12OL 23518511 IC50 = 80 nM T47101 CRX0Q6 23625758 IC50 = 400 nM T47101 C2RV3U 24180608 IC50 = 9700 nM T47101 CQNP54 24764449 IC50 = 25000 nM T47101 C81GVC 24774737 IC50 < 15.85 nM T47101 CN6B1L 24774912 IC50 = 25.12 nM T47101 CAO30M 24775639 IC50 = 100 nM T47101 CFK2B9 24882503 IC50 = 570 nM T47101 C43HWQ 24883287 IC50 > 10000 nM T47101 C8DA5Q 24883334 IC50 > 10000 nM T47101 C0P6AU 24894017 IC50 = 3340 nM T47101 CY8L7E 24896769 IC50 > 10000 nM T47101 C15BZP 24949852 IC50 = 560 nM T47101 CZHE50 24949856 IC50 = 600 nM T47101 C9YN2Q 24967131 IC50 > 10000 nM T47101 C4EG8R 24993189 IC50 > 10000 nM T47101 CN3FQ5 25014760 IC50 = 183 nM T47101 C3WX2S 25014762 IC50 = 313 nM T47101 C3SE8L 25014843 IC50 = 112 nM T47101 CV0RN4 25014844 IC50 = 738 nM T47101 CZ8LP3 25014846 IC50 = 501 nM T47101 CO0R9B 25014936 IC50 = 1580 nM T47101 CRA79I 25015025 IC50 = 56 nM T47101 CGDP84 25015026 IC50 = 447 nM T47101 CSD14Z 25015027 IC50 = 1550 nM T47101 C0HVE3 25015107 IC50 = 350 nM T47101 CV67GQ 25015556 IC50 = 720 nM T47101 CTV54O 25123227 IC50 = 2700 nM T47101 CTED51 25186142 IC50 = 1.995 nM T47101 C8YLD6 25194331 IC50 = 30 nM T47101 CXC9B3 25194865 IC50 = 370 nM T47101 C1I0VS 25194866 IC50 = 110 nM T47101 C9OZN3 25194867 IC50 = 1800 nM T47101 CNG96H 25210579 IC50 > 10000 nM T47101 CVM13K 42596931 IC50 = 178 nM T47101 C92RQB 42600929 IC50 = 114.5 nM T47101 C8T5IH 42602949 IC50 = 5.012 nM T47101 CKO7F0 42645244 IC50 = 1380 nM T47101 C0C1HL 42645248 IC50 = 998 nM T47101 CS3AI0 42645478 IC50 = 140 nM T47101 CN8WB9 44189332 IC50 = 175 nM T47101 CEL61X 44229839 IC50 > 10000 nM T47101 CHZ6Q1 44269004 IC50 = 17100 nM T47101 CH3J2E 44299176 IC50 = 200 nM T47101 C27GVO 44299203 IC50 = 400 nM T47101 CY6WC0 44299236 IC50 = 400 nM T47101 C3RG0C 44299304 IC50 = 500 nM T47101 CJM26I 44299321 IC50 = 3400 nM T47101 C9UGL3 44299325 IC50 = 1200 nM T47101 CJEZ96 44299338 IC50 = 1100 nM T47101 C8XGN5 44299339 IC50 = 80 nM T47101 CNH34G 44299354 IC50 = 600 nM T47101 C82MSD 44299360 IC50 = 1700 nM T47101 CYV2D7 44368815 IC50 = 5100 nM T47101 CWR4Q0 44398656 IC50 = 260 nM T47101 CUA37S 44398657 IC50 = 330 nM T47101 CZ7TN1 44398732 IC50 = 190 nM T47101 C8K4AL 44407237 IC50 > 50000 nM T47101 CUA18B 44407238 IC50 = 23600 nM T47101 C04HFE 44407248 IC50 > 50000 nM T47101 CR3O1C 44407275 IC50 = 8800 nM T47101 C70BFV 44407276 IC50 = 38400 nM T47101 CMH7W6 44407277 IC50 = 23800 nM T47101 CETQ79 44427518 IC50 > 50000 nM T47101 COPG94 44427519 IC50 > 10000 nM T47101 CUB12D 44449577 IC50 = 61 nM T47101 C4WRN5 44541014 IC50 = 50 nM T47101 C3VRO9 44557921 IC50 > 10000 nM T47101 C3HW7L 44570553 IC50 > 30000 nM T47101 C17PVE 44570554 IC50 > 30000 nM T47101 CLOY92 44570599 IC50 = 2000 nM T47101 CK06LT 44570600 IC50 > 30000 nM T47101 CXD9B4 44578561 IC50 = 2900 nM T47101 CPUB89 45103791 IC50 = 250000 nM T47101 CQC29U 45103904 IC50 = 4000 nM T47101 CUQL91 45103905 IC50 = 5500 nM T47101 CP2YM3 45103907 IC50 = 1900 nM T47101 CU3RF1 45139989 IC50 > 10000 nM T47101 CQGZ06 45139991 IC50 > 10000 nM T47101 C4KWJ3 45379956 IC50 = 18060 nM T47101 C2CU0B 45380067 IC50 = 28790 nM T47101 C4QK2M 46182943 IC50 > 10000 nM T47101 CMB71C 46182945 IC50 = 65 nM T47101 CV45ZD 46182946 IC50 = 77 nM T47101 CP7T6B 46182947 IC50 > 10000 nM T47101 C8S2KY 46182948 IC50 = 577 nM T47101 CEUW42 46183177 IC50 > 10000 nM T47101 CJXD56 46183178 IC50 = 424 nM T47101 CG74EC 46186409 IC50 > 10000 nM T47101 C2GI4X 46186410 IC50 > 10000 nM T47101 CUP02A 46186412 IC50 > 10000 nM T47101 CWF9N5 46186413 IC50 > 10000 nM T47101 CO60DU 46186664 IC50 > 10000 nM T47101 C9T5AS 46186665 IC50 > 10000 nM T47101 CZ6D3F 46186666 IC50 = 3600 nM T47101 C5YK9M 46186668 IC50 = 19 nM T47101 CKSC63 46186670 IC50 > 10000 nM T47101 CY3HW5 46224684 IC50 > 10000 nM T47101 C2P9QO 46228508 IC50 > 10000 nM T47101 C6E5PY 46228822 IC50 = 4250 nM T47101 C3T8AM 46228951 IC50 > 10000 nM T47101 C7ON5A 46233287 IC50 > 10000 nM T47101 CSLY07 46233305 IC50 = 3300000 nM T47101 C9H4YO 46233889 IC50 = 200 nM T47101 CRT34L 46235770 IC50 = 11 nM T47101 C0WYM1 46898022 IC50 = 10000 nM T47101 CHSF07 49806372 IC50 > 1000 nM T47101 C9L3XR 49838879 IC50 > 50000 nM T47101 CF91RS 49843531 IC50 > 10000 nM T47101 CB5O0I 49860186 IC50 = 1500 nM T47101 C9W6SO 49860190 IC50 = 2000 nM T47101 C2Y6QS 50938552 IC50 > 10000 nM T47101 C90ANW 50939489 IC50 = 18 nM T47101 CS9G6E 50997096 IC50 > 10000 nM T47101 C9NYP4 51036677 IC50 > 10000 nM T47101 C4WRY3 51037112 IC50 > 10000 nM T47101 CRI28Z 51037948 IC50 > 10000 nM T47101 CVZU97 51346202 IC50 = 840 nM T47101 CTC8N1 51352971 IC50 = 26 nM T47101 C5QK8Y 51352972 IC50 = 760 nM T47101 CL4I2K 52941234 IC50 = 27000 nM T47101 C7S9UY 52941519 IC50 = 4500 nM T47101 C39IPC 52942177 IC50 = 270 nM T47101 CN3H2J 52942791 IC50 = 220 nM T47101 CSG8U1 52943668 IC50 > 10000 nM T47101 C6R8AL 52943750 IC50 > 10000 nM T47101 CH3FO1 52943828 IC50 > 10000 nM T47101 CB56DX 52943829 IC50 = 940 nM T47101 CKP62L 52944574 IC50 > 10000 nM T47101 CIB62R 52944613 IC50 > 10000 nM T47101 C4R3IB 52944922 IC50 > 10000 nM T47101 CUDK18 52945153 IC50 = 610 nM T47101 CZNE23 52945805 IC50 = 14 nM T47101 C6OI2Q 52946085 IC50 > 10000 nM T47101 CU4Q1F 52946141 IC50 > 10000 nM T47101 C95BXO 52946218 IC50 > 10000 nM T47101 C17KVM 52946496 IC50 = 6500 nM T47101 C57VIC 52947692 IC50 = 390 nM T47101 C63VCY 52948336 IC50 > 10000 nM T47101 CIPT89 52948377 IC50 > 10000 nM T47101 CNZ0E5 52948579 IC50 > 10000 nM T47101 CE3WD7 52948666 IC50 > 10000 nM T47101 CIKY86 52949957 IC50 = 260 nM T47101 CL7K3V 52949960 IC50 > 10000 nM T47101 C09SDH 53257410 IC50 = 74 nM T47101 CS64CJ 53257411 IC50 = 485 nM T47101 CGEU76 53257412 IC50 = 216 nM T47101 C7DTK5 53259208 IC50 > 10000 nM T47101 CZ48HC 53259209 IC50 > 10000 nM T47101 CW1DS4 53259393 IC50 = 2100 nM T47101 CM89OC 53259394 IC50 = 320 nM T47101 C31PHF 53259395 IC50 > 10000 nM T47101 C2SZ0F 53259396 IC50 > 10000 nM T47101 C4YF9G 53259397 IC50 > 10000 nM T47101 CNPM14 53341082 IC50 > 3000 nM T47101 C4F6SR 53348188 IC50 = 3.6 nM T47101 CBK9Q6 53357848 IC50 > 10000 nM T47101 C8NA4L 53384644 IC50 > 30000 nM T47101 CVG90B 53389651 IC50 > 10000 nM T47101 C04YJS 53408448 IC50 = 90000 nM T47101 CA7W1M 54582410 IC50 = 4500 nM T47101 CO6B0E 54583043 IC50 > 10000 nM T47101 C3PGE2 54585958 IC50 > 10000 nM T47101 CV7HJ8 54585959 IC50 > 10000 nM T47101 C47JTI 54586838 IC50 = 662 nM T47101 CE1ZK6 54759168 IC50 > 10000 nM T47101 C8AB1J 54759606 Ki = 350 nM T47101 CCR36T 55264593 IC50 = 77000 nM T47101 CM8JX1 56604907 IC50 = 1000 nM T47101 C9DX3J 56649281 IC50 = 26 nM T47101 CBOD63 56835089 IC50 > 30000 nM T47101 CR50TJ 56835147 IC50 > 10000 nM T47101 CY36EG 56945171 IC50 = 1600 nM T47101 C4OG7H 56945172 IC50 = 2800 nM T47101 CH0QA3 56945173 IC50 = 1000 nM T47101 CM0NQ5 56945174 IC50 = 2000 nM T47101 CXKF03 56945175 IC50 = 4100 nM T47101 C6WU4V 56945277 IC50 = 12 nM T47101 CAK91L 56955954 IC50 > 3600 nM T47101 CDS06V 56973548 IC50 = 501.19 nM T47101 CUAV97 56973549 IC50 = 63.1 nM T47101 CI0K7Y 56973550 IC50 = 63.1 nM T47101 CD6Y9Z 57395116 IC50 > 30000 nM T47101 C8W6IG 57395117 IC50 = 22700 nM T47101 CG7S0D 57396882 IC50 > 30000 nM T47101 C8P6RD 57505528 IC50 = 5100 nM T47101 CPU2E3 59737752 IC50 = 6350 nM T47101 C1MR8Q 60097495 IC50 > 1000 nM T47101 COM48T 60154284 IC50 = 630.96 nM T47101 CB7KE0 60154285 IC50 = 63.1 nM T47101 CO75BK 60154286 IC50 = 31.62 nM T47101 CEF48W 60154326 IC50 = 100 nM T47101 C2Y7JC 60154327 IC50 = 31.62 nM T47101 COU2B3 60154328 IC50 = 79.43 nM T47101 CKM5E6 60154329 IC50 = 79.43 nM T47101 CVE49A 60154330 IC50 = 7.943 nM T47101 C3BMS1 60154331 IC50 = 199.53 nM T47101 CBU4I5 60154332 IC50 = 125.89 nM T47101 C03CFA 60154333 IC50 = 199.53 nM T47101 CLK0O6 60154334 IC50 = 100 nM T47101 C34QJR 60154335 IC50 = 398.11 nM T47101 CXO1I8 60154336 IC50 = 79.43 nM T47101 CNZX63 60154337 IC50 = 5011.87 nM T47101 C3I4KJ 60154338 IC50 = 100 nM T47101 CRB5D8 60154339 IC50 = 794.33 nM T47101 CYI9F7 60154340 IC50 = 39.81 nM T47101 CLY46E 60154341 IC50 = 79.43 nM T47101 CNS3Y1 60154342 IC50 = 25.12 nM T47101 C7CS4I 60154343 IC50 = 63.1 nM T47101 C46LSW 60154344 IC50 = 25.12 nM T47101 CR60YI 60154345 IC50 = 63.1 nM T47101 CSZA16 60155724 IC50 > 3600 nM T47101 CU79HD 60202383 IC50 = 63 nM T47101 C9ZCT2 62705065 IC50 > 1000 nM T47101 C10AMI 66553589 IC50 = 3480 nM T47101 C9O4GF 66555232 IC50 = 2.9 nM T47101 CBA0S2 66555775 IC50 = 6000 nM T47101 CL3EN2 66556938 IC50 = 49 nM T47101 C9QF6B 66559005 IC50 = 63 nM T47101 CE49GC 67098566 Ki = 80 nM T47101 C37NKO 67129970 IC50 > 10000 nM T47101 CK80LJ 67130050 IC50 > 10000 nM T47101 CQ97ZW 67161103 IC50 = 12 nM T47101 CNP52W 67163022 IC50 = 13 nM T47101 CV63UL 67240318 IC50 > 5000 nM T47101 CO6W9D 68004741 IC50 = 1.5 nM T47101 CB6U7F 68005465 IC50 = 2.9 nM T47101 CK83VI 68005486 IC50 = 50 nM T47101 C1RJ7Y 68005600 IC50 = 56 nM T47101 COX3U9 68005621 IC50 = 3 nM T47101 CEXN58 68005732 IC50 = 33 nM T47101 C8I7GC 68293638 IC50 > 10000 nM T47101 C7GRV2 68755406 IC50 > 10000 nM T47101 CEBO91 71452977 IC50 > 10000 nM T47101 CCN01X 71547862 IC50 > 10000 nM T47101 C1NPL0 71552941 IC50 > 30000 nM T47101 CA4PS8 71552942 IC50 > 30000 nM T47101 C3UA9C 71553011 IC50 = 30000 nM T47101 CEZ15Y 71553012 IC50 = 12510 nM T47101 CVIA91 71553085 IC50 = 30000 nM T47101 C1TR3O 71553152 IC50 = 30000 nM T47101 CN7W5S 71579325 IC50 > 10000 nM T47101 C1BCX0 71579696 IC50 > 1000 nM T47101 CZ31PU 71583657 IC50 > 10000 nM T47101 CU1IL6 71741204 IC50 > 100000 nM T47101 CN1GA3 71741327 IC50 > 100000 nM T47101 COS5D7 71741328 IC50 > 100000 nM T47101 C8PWZ0 71741329 IC50 > 100000 nM T47101 CT4XR9 71741332 IC50 > 100000 nM T47101 C9OQ2I 72710839 IC50 = 239.9 nM T47101 C60TUV 72737208 IC50 > 10000 nM T47101 CJ3WA6 72737404 IC50 > 10000 nM T47101 C6R8DI 72943374 IC50 = 145 nM T47101 CV21FR 73349643 IC50 = 5000 nM T47101 C9TMA1 73352657 IC50 = 4200 nM T47101 CYQ8K1 73357210 IC50 = 900 nM T47101 CVNW01 73386831 IC50 > 1000 nM T47101 CQ5E3H 73707531 IC50 = 1 nM T47101 CGDB30 74538658 IC50 = 250 nM T47101 C47HYO 76329677 IC50 > 20000 nM T47101 C3DF1L 86278931 IC50 = 1.4 nM T47101 C0GQ8S 86291490 IC50 = 1.2 nM T47101 C25LFJ 86291934 IC50 = 2.1 nM T47101 CQ7DT9 86291937 IC50 = 0.8 nM T47101 CZE71X 86292511 IC50 = 0.2 nM T47101 C8DLZ9 86292714 IC50 = 1.1 nM T47101 CU6IH5 86292906 IC50 = 1 nM T47101 C40UFG 86292907 IC50 = 4.7 nM T47101 CKP0G4 86292908 IC50 = 0.8 nM T47101 CO0XH6 86293092 IC50 = 37 nM T47101 CRQO23 86293280 IC50 = 250 nM T47101 C4OC7T 86293469 IC50 = 38 nM T47101 CV5R1Q 86293660 IC50 = 2.8 nM T47101 CP3E7G 86293661 IC50 = 1.3 nM T47101 C2XVA8 86293662 IC50 = 1.9 nM T47101 CWG2N9 86293663 IC50 = 1.6 nM T47101 C5G6OD 86293664 IC50 = 4.7 nM T47101 CPU6V0 86293851 IC50 = 9.4 nM T47101 C2AMK8 86293852 IC50 = 5.3 nM T47101 C2MIB0 86294035 IC50 = 24 nM T47101 CURD29 86294412 IC50 = 1.3 nM T47101 CUR3G0 86294415 IC50 = 1.5 nM T47101 CCJ43A 86302281 IC50 > 10000 nM T47101 CB5NJ4 86302541 IC50 = 643.7 nM T47101 CPG3A5 86302574 IC50 > 30000 nM T47101 CWZ41G 86566934 IC50 = 12.8 nM T47101 C0ALG3 86567077 IC50 = 7.6 nM T47101 CW40TZ 86567079 IC50 = 5.7 nM T47101 CEY30N 86567080 IC50 = 3 nM T47101 C3I5JQ 86567457 IC50 = 1.1 nM T47101 C1BZA4 86567460 IC50 = 6.7 nM T47101 C5S7BY 86567464 IC50 = 1.1 nM T47101 C5F7IL 86567465 IC50 > 100 nM T47101 C35KFO 86567537 IC50 > 100 nM T47101 CN48JU 86567539 IC50 > 100 nM T47101 C1Z8UJ 86567604 IC50 = 1.3 nM T47101 CZ0L3H 86567605 IC50 = 5.2 nM T47101 CGA10Z 86567606 IC50 = 26.5 nM T47101 C0K2VG 86567607 IC50 = 8.1 nM T47101 C07KPY 86567668 IC50 = 11.2 nM T47101 C1C5PN 86567669 IC50 = 1.6 nM T47101 CLO6A7 86567670 IC50 = 2.2 nM T47101 CR1N0E 90367910 IC50 = 0.5 nM T47101 CFB75T 90479825 IC50 = 160 nM T47101 CY0UC4 90645194 IC50 > 10000 nM T47101 C3GU7P 90645237 IC50 > 10000 nM T47101 CFI93O 90645239 IC50 > 10000 nM T47101 C76KSB 90645241 IC50 > 10000 nM T47101 CNWP80 90645243 IC50 > 10000 nM T47101 C1POJ2 90645244 IC50 > 10000 nM T47101 C8BEX4 90645245 IC50 > 10000 nM T47101 CX29IY 90655145 IC50 > 10000 nM T47101 CA6Q1I 91801169 IC50 = 15 nM T47101 CF27DP 91825767 IC50 = 1 nM T47101 C4CE3S 94146587 IC50 = 57150 nM T47101 CN2XT7 117703686 IC50 = 1.6 nM T47101 CI5LW2 117715251 IC50 = 13 nM T47101 CR9S7W 118036565 IC50 > 10000 nM T47101 CUTW04 118036840 IC50 > 10000 nM T47101 C0ZUO9 118295608 IC50 = 1.8 nM T47101 C0P6JC 118295611 IC50 = 1 nM T47101 COZU45 118295731 IC50 = 0.4 nM T47101 C49VZY 118295741 IC50 = 4.1 nM T47101 CZ0X2U 118295886 IC50 = 11 nM T47101 C5JDF9 118296035 IC50 = 0.7 nM T47101 CY7BI2 118706214 IC50 > 10000 nM T47101 CVB8Q7 118728412 IC50 = 20 nM T47101 CQML87 118728663 IC50 = 450 nM T47101 CX1IU7 118753064 IC50 > 30000 nM T47101 CI93JD 118893305 IC50 = 0.3 nM T47101 CH1B5J 118893306 IC50 = 0.3 nM T47101 CN9PU5 118893320 IC50 = 7.7 nM T47101 C9WY7M 118893324 IC50 = 6.2 nM T47101 CMY9G2 118893337 IC50 = 0.5 nM T47101 C2PY9L 118893647 IC50 = 3.3 nM T47101 CEQH07 122378841 IC50 = 5200 nM T47101 C7E5HN 122378842 IC50 > 20000 nM T47101 CLM7K3 122604539 IC50 = 3500 nM T47101 C01JHI 122604566 IC50 = 8600 nM T47101 C1E4AR 122604567 IC50 = 4340 nM T47101 CQJZ70 122604640 IC50 = 2900 nM T47101 CMQ9V3 122606542 IC50 = 60 nM T47101 CY30FL 123752658 IC50 = 0.5 nM T47101 C6PQI0 126481264 IC50 = 228.2 nM T47101 CO81RL 126481269 IC50 = 5.1 nM T47101 CUF81C 127025156 IC50 > 500 nM T47101 CP3LK5 127025157 IC50 = 28.23 nM T47101 C8QKX6 127025158 IC50 = 104.2 nM T47101 CDQ52G 127025443 IC50 = 69.34 nM T47101 C8KXV1 127025843 IC50 > 1000 nM T47101 CBT52X 127027296 IC50 > 500 nM T47101 CS6TJ8 127027297 IC50 = 129.86 nM T47101 C0EZA2 127027298 IC50 > 500 nM T47101 CER0Q3 127027305 IC50 = 99.15 nM T47101 CAH9J6 127027306 IC50 > 500 nM T47101 CN3SW5 127027307 IC50 > 500 nM T47101 CC0R4L 127027308 IC50 = 96.15 nM T47101 C7EYC2 127027620 IC50 = 81.28 nM T47101 C12ODR 127027621 IC50 = 271.85 nM T47101 CA7JW5 127027622 IC50 > 500 nM T47101 CMT3C7 127027623 IC50 > 500 nM T47101 C0T3HO 127027641 IC50 > 500 nM T47101 CLO6P4 127027642 IC50 = 260.79 nM T47101 CKS28E 127034802 IC50 > 1000 nM T47101 CWRB15 127034986 IC50 = 154.16 nM T47101 CM09WL 127035009 IC50 = 32.57 nM T47101 CDU87A 127035163 IC50 = 370.6 nM T47101 CO26SA 127036029 IC50 > 20000 nM T47101 CEPL09 127036182 IC50 > 500 nM T47101 C87BIU 127036183 IC50 = 99.75 nM T47101 CR0NI6 127036477 IC50 = 333.89 nM T47101 CM17TO 127036596 IC50 = 56.49 nM T47101 C52JBY 127036758 IC50 > 500 nM T47101 C72EXH 127036764 IC50 = 138.06 nM T47101 CKX40V 127037812 IC50 > 10000 nM T47101 C70RUP 127038480 IC50 > 10000 nM T47101 C3WCN8 127041777 IC50 > 10000 nM T47101 CHK16Q 127045929 IC50 > 1000 nM T47101 CY3J0C 127047591 IC50 > 1000 nM T47101 C9SI5T 127047969 IC50 < 0.2 nM T47101 CTS97V 129308354 IC50 = 11.7 nM T47101 C0FM1R 130196825 IC50 > 30000 nM T47101 C8ARK0 131801160 IC50 = 54 nM T47101 C9Y5TL 132156608 IC50 > 10000 nM T47101 CUO0C5 132156633 IC50 > 10000 nM T47101 CUW5L2 132156656 IC50 > 10000 nM T47101 CT3DM9 132156669 IC50 > 10000 nM T47101 CY35PA 132156727 IC50 > 10000 nM T47101 C0R2MF 132156728 IC50 > 10000 nM T47101 CZN5W1 132156731 IC50 > 10000 nM T47101 CQB04N 132156743 IC50 > 10000 nM T47101 C53HPM 132156749 IC50 > 10000 nM T47101 C3UA1J 132156758 IC50 > 10000 nM T47101 CJ7B4Q 132156777 IC50 > 10000 nM T47101 C8A7XK 132156780 IC50 > 10000 nM T47101 CBWE03 132156803 IC50 > 10000 nM T47101 CO3P6X 132156815 IC50 > 10000 nM T47101 C95HIB 132156818 IC50 > 10000 nM T47101 C3CD6R 132156853 IC50 > 10000 nM T47101 CML72V 132185297 IC50 = 0.8 nM T47101 CM8TC3 132185299 IC50 = 30.9 nM T47101 CWY58Z 132185302 Ki = 10 nM T47101 CQL4B7 132185442 IC50 = 10.8 nM T47101 C3V5TF 132245876 IC50 > 100 nM T47101 CXA84S 132245879 IC50 = 0.3 nM T47101 C8HPV6 132245890 IC50 < 0.3 nM T47101 C4F9YW 132245892 IC50 = 0.6 nM T47101 C5QZ7A 132245893 IC50 = 0.8 nM T47101 CA3IV9 132245894 IC50 = 2.9 nM T47101 C95XEY 132245912 IC50 = 30.9 nM T47101 CIJ6Y0 132245918 IC50 = 9 nM T47101 CKW5S9 132245920 IC50 = 163.9 nM T47101 CX3ZV1 132245921 IC50 = 2.6 nM T47101 C8U1MG 132245924 IC50 = 1.4 nM T47101 C6H3JS 132245929 IC50 = 0.8 nM T47101 CPN39H 132245933 IC50 = 2.5 nM T47101 C8U0OD 132245935 IC50 = 0.8 nM T47101 C7VW5M 132245939 IC50 < 0.3 nM T47101 CMER63 132245964 IC50 = 2.6 nM T47101 CRIN01 132245965 IC50 = 0.6 nM T47101 C5XLN0 132245967 IC50 = 2.1 nM T47101 CFY9W5 132245971 IC50 = 7.2 nM T47101 CULE97 132245973 IC50 = 40.3 nM T47101 C5K7YE 132246005 IC50 = 105.1 nM T47101 CR85IS 132246032 IC50 = 4.4 nM T47101 C2JPX7 132246037 IC50 = 3.8 nM T47101 C4YSB5 132246051 IC50 = 0.8 nM T47101 CERS64 132937256 IC50 > 30000 nM T47101 CK9W4F 134135741 IC50 = 1900 nM T47101 CMA60G 134144799 IC50 > 50000 nM T47101 C3MN6B 134144868 IC50 = 1100 nM T47101 CEZH84 134146580 IC50 = 160 nM T47101 C1DF4R 134147544 IC50 = 450 nM T47101 C95NCV 134151662 IC50 = 130 nM T47101 CX7YE1 134155961 IC50 = 69 nM T47101 CE38MW 134156584 IC50 = 1.2 nM T47101 CVI25K 134157526 IC50 = 270 nM T47101 C71CBJ 134255819 IC50 > 10000 nM T47101 CBGO29 134255820 IC50 > 10000 nM T47101 CI8L9W 134255882 IC50 > 10000 nM T47101 C5UBG7 134255896 IC50 > 10000 nM T47101 CVE4X3 134457519 IC50 > 10000 nM T47101 CO1IL0 134457555 IC50 > 10000 nM T47101 CB15KN 134457556 IC50 > 10000 nM T47101 CCFS35 134457606 IC50 > 10000 nM T47101 CEAH09 134457612 IC50 > 10000 nM T47101 C1P9KY 134457618 IC50 > 10000 nM T47101 CGAV72 134457621 IC50 = 617.7 nM T47101 CJYX87 134457890 IC50 > 10000 nM T47101 C2AN7T 134611886 IC50 > 100000 nM T47101 CYL5V1 134694986 IC50 > 30000 nM T47101 CWZ1L4 135316948 IC50 = 0.91 nM T47101 C5B6XD 135316952 IC50 = 1.32 nM T47101 CUE8M0 135316960 IC50 = 4.59 nM T47101 CWEP52 135316962 IC50 = 1.16 nM T47101 CW5KL0 135316982 IC50 = 1.07 nM T47101 C6E5FP 135317017 IC50 = 0.28 nM T47101 CSB6A4 135317061 IC50 = 3.08 nM T47101 CMT6S2 135317122 IC50 = 1.81 nM T47101 CCTW97 135317286 IC50 = 1.06 nM T47101 CFV71G 135317433 IC50 = 2.28 nM T47101 CH2JK6 135317468 IC50 = 1.18 nM T47101 C7E0VW 135317479 IC50 = 1.77 nM T47101 C9M3AS 135317507 IC50 = 2.33 nM T47101 CD24PG 135317520 IC50 = 1.97 nM T47101 CFE0X7 135317546 IC50 = 0.73 nM T47101 C0JM1W 135317567 IC50 = 1.21 nM T47101 C12QZN 135317616 IC50 = 10.7 nM T47101 CI2L5A 135317791 IC50 = 0.99 nM T47101 CJZ59L 135317844 IC50 = 1.06 nM T47101 C45XNW 135318783 IC50 = 1.23 nM T47101 CLCO61 135398510 IC50 = 8 nM T47101 CLSE63 135398512 IC50 = 28 nM T47101 CB8GH1 135398810 IC50 > 30000 nM T47101 C2TPB3 135398811 IC50 > 30000 nM T47101 C2C3JF 135398812 IC50 = 10000 nM T47101 CL3J2V 135398815 IC50 = 1120 nM T47101 C7TQC8 135398816 IC50 > 30000 nM T47101 C78NHD 135398825 IC50 = 3500 nM T47101 CBV73N 135398830 IC50 = 600 nM T47101 C5LYR7 135398831 IC50 > 30000 nM T47101 CY58IA 135398833 IC50 > 30000 nM T47101 CRP0M1 135398834 IC50 = 3280 nM T47101 CX82YT 135400685 IC50 = 7000 nM T47101 CN5T7W 135400982 IC50 = 70 nM T47101 CVJ07T 135402853 IC50 = 390 nM T47101 C76JPR 135405015 IC50 = 5 nM T47101 CBK6I2 135407156 IC50 = 80 nM T47101 CMVS34 135410282 IC50 = 44 nM T47101 C34FSG 135410286 IC50 = 576 nM T47101 CYQG80 135417125 IC50 = 27000 nM T47101 CUT52Q 135421574 IC50 > 25000 nM T47101 CW85GB 135426457 IC50 = 9900 nM T47101 CV8Q7A 135430397 IC50 = 11 nM T47101 C8X5SV 135433815 IC50 = 90 nM T47101 CO15RE 135435545 IC50 > 30000 nM T47101 CM4J6A 135444580 IC50 = 50 nM T47101 CNZ04G 135453357 IC50 = 20 nM T47101 C1M3PW 135458467 IC50 = 20.3 nM T47101 CS63IO 135476717 IC50 = 69 nM T47101 C9D2FL 135483378 IC50 > 4880 nM T47101 C4WX3I 135486449 IC50 = 15180 nM T47101 CA80OZ 135488014 IC50 = 5 nM T47101 CDCF48 135488027 IC50 = 14 nM T47101 CUDY67 135491327 IC50 > 30000 nM T47101 C69FTB 135496141 IC50 = 3000 nM T47101 CG5HY4 135507297 IC50 = 10 nM T47101 CT0NV5 135514617 IC50 = 20 nM T47101 C57FTA 135527773 IC50 = 28200 nM T47101 CM6W4K 135527782 IC50 = 11000 nM T47101 CK8TR4 135527783 IC50 = 7300 nM T47101 CFPV27 135543821 IC50 = 50 nM T47101 CRCH86 135546221 IC50 = 1010 nM T47101 C65XMQ 135546228 IC50 = 8 nM T47101 CMT3X5 135584854 IC50 = 2120 nM T47101 CW08GF 135674125 IC50 = 390 nM T47101 CLS64T 135674129 IC50 = 550 nM T47101 C54ABM 135674133 IC50 = 1 nM T47101 CM7YH4 135674136 IC50 = 20 nM T47101 C1WSO7 135674140 IC50 = 4100 nM T47101 CA0Y7V 135674142 IC50 = 20 nM T47101 CM90FP 135674144 IC50 = 10 nM T47101 C3CP1X 135674147 IC50 = 2 nM T47101 CBSV42 135674149 IC50 = 21 nM T47101 C1NTB0 135674153 IC50 = 8 nM T47101 CID0W9 135674167 IC50 = 1 nM T47101 C1DL9J 135674173 IC50 = 120 nM T47101 CO89UX 135674193 IC50 = 24 nM T47101 CSB6O2 135738245 IC50 = 2280 nM T47101 CT6Q0X 135738246 IC50 = 320 nM T47101 C7N3PA 135773881 IC50 = 1850 nM T47101 CT62ND 135773888 IC50 = 630 nM T47101 CH2R9N 135773902 IC50 = 27000 nM T47101 C0PVG7 135819982 IC50 = 1 nM T47101 CQ92DH 135819983 IC50 = 16 nM T47101 C9ZI5J 135820026 IC50 = 15 nM T47101 C9LG3C 135820141 IC50 = 18 nM T47101 CWI61Y 135820280 IC50 = 94 nM T47101 C53LFX 135820297 IC50 = 8 nM T47101 CM2AO1 135820333 IC50 = 100 nM T47101 C5BI9T 135820431 IC50 = 23 nM T47101 CYHV16 135820505 IC50 = 830 nM T47101 CXJ19P 135839366 IC50 = 2660 nM T47101 C0QH5E 135839368 IC50 = 100 nM T47101 C01OLI 135839369 IC50 = 3170 nM T47101 CP1H7K 135839370 IC50 = 5000 nM T47101 C2PIQ9 135839371 IC50 = 43 nM T47101 CK6H2P 135839372 IC50 = 348 nM T47101 C2H3XB 135926086 IC50 = 9 nM T47101 C7BES6 135926087 IC50 = 15 nM T47101 CNTK81 135926088 IC50 = 7 nM T47101 CQ64OH 135926089 IC50 = 900 nM T47101 CXG7O4 135926090 IC50 = 10 nM T47101 CN4FG3 135926091 IC50 = 190 nM T47101 C7NZU3 135926094 IC50 > 25000 nM T47101 CL6HQ4 135926104 IC50 = 3 nM T47101 CE37KQ 135926113 IC50 = 3 nM T47101 C1ZRT7 135926114 IC50 = 40 nM T47101 CU5W2V 135926115 IC50 = 83 nM T47101 C1D3EW 135926116 IC50 = 8 nM T47101 CXM75Z 135985610 IC50 = 13 nM T47101 CHA4N2 136013680 IC50 > 10 nM T47101 C23SGN 136038438 IC50 = 200 nM T47101 CS91JC 136038439 IC50 = 2 nM T47101 C5DVE4 136038477 IC50 > 3000 nM T47101 CAG34B 136038492 IC50 = 270 nM T47101 C7Q1KT 136038570 IC50 > 3000 nM T47101 C9SL4U 136038593 IC50 = 3 nM T47101 CAXJ50 136043793 IC50 = 48 nM T47101 CF12ME 136043801 IC50 = 73 nM T47101 CE4Y0B 136043806 IC50 = 210 nM T47101 C7JF8X 136043808 IC50 = 98 nM T47101 CTAY92 136043832 IC50 = 82 nM T47101 C1V8PI 136087061 IC50 = 1200 nM T47101 CU05YS 136118622 IC50 = 326 nM T47101 CN49OS 136118623 IC50 = 199 nM T47101 C39CXW 136118624 IC50 = 70 nM T47101 CR48NF 136118625 IC50 = 300 nM T47101 CD5M9T 136118626 IC50 = 287 nM T47101 CW27AO 136118641 IC50 = 1950 nM T47101 CZHA29 136118700 IC50 = 205 nM T47101 CFD03R 136118701 IC50 = 814 nM T47101 C3SIK1 136118702 IC50 = 187 nM T47101 C4LC2Q 136118703 IC50 = 950 nM T47101 CX39CA 136118704 IC50 = 79 nM T47101 C3PI2X 136118707 IC50 = 4000 nM T47101 C2OAK8 136118708 IC50 = 628 nM T47101 C6PUG0 136118709 IC50 = 4899 nM T47101 CH1E7I 136118710 IC50 = 725 nM T47101 C0RBJ7 136118711 IC50 = 86 nM T47101 C4V8HY 136118712 IC50 = 6293 nM T47101 CZ4AF8 136118717 IC50 = 57 nM T47101 CMP78A 136118718 IC50 = 446 nM T47101 CN8RB4 136118719 IC50 = 4880 nM T47101 CIUJ95 136118720 IC50 = 4880 nM T47101 C2BIZ5 136118721 IC50 = 75 nM T47101 C5YL7I 136118722 IC50 = 1586 nM T47101 CZQ5P1 136118733 IC50 = 24400 nM T47101 CMP4R8 136118734 IC50 = 67 nM T47101 C7E6XJ 136118735 IC50 = 51 nM T47101 CCX81R 136118736 IC50 = 39 nM T47101 C29ZXF 136118737 IC50 = 42 nM T47101 C5QZ4H 136126664 IC50 = 7900 nM T47101 CB8RX0 136126665 IC50 = 190 nM T47101 CYXU86 136180312 IC50 = 9590 nM T47101 C9MHA4 136180313 IC50 = 4840 nM T47101 C2OQ8Z 136211076 IC50 = 1.4 nM T47101 CDT7E4 136211077 IC50 = 0.9 nM T47101 C2ARQ5 136211078 IC50 = 20.8 nM T47101 C71KBR 136211079 IC50 = 6.6 nM T47101 C8LMA2 136211080 IC50 = 2.7 nM T47101 CO4WD5 136211081 IC50 = 22.4 nM T47101 C1YUD0 136219394 IC50 > 10 nM T47101 C7PNC4 136243300 IC50 = 15220 nM T47101 CUN1I4 136243344 IC50 = 12650 nM T47101 C68IKN 136243473 IC50 = 11910 nM T47101 CIU8W3 136254389 IC50 > 10 nM T47101 CE7L0G 136269119 IC50 = 18325 nM T47101 C7U9GP 136269138 IC50 = 33849 nM T47101 C35MBU 136299423 IC50 = 140 nM T47101 C0W8KA 136299435 IC50 = 120 nM T47101 C5G4ES 136299436 IC50 = 100 nM T47101 CDY18N 136301774 IC50 = 12000 nM T47101 C1VDW4 136380921 IC50 = 3800 nM T47101 CH4T8M 136961363 IC50 = 5330 nM T47101 C7N8EG 136961364 IC50 = 17840 nM T47101 CRPQ98 136961365 IC50 = 15040 nM T47101 CSZ16N 136961366 IC50 = 9130 nM T47101 CB9D7F 136961367 IC50 = 3170 nM T47101 CEPT42 136961368 IC50 = 1560 nM T47101 C3QY0H 137133096 IC50 > 1000 nM T47101 C59TAF 137133097 IC50 = 9.4 nM T47101 CZB0G9 137133098 IC50 = 13.6 nM T47101 C28OFT 137133102 IC50 = 2.1 nM T47101 C09POL 137133106 IC50 = 0.3 nM T47101 CL4M3P 137133110 IC50 = 1.5 nM T47101 CNUX28 137133111 IC50 = 0.4 nM T47101 CNH5T6 137133114 IC50 = 2.1 nM T47101 CXR23D 137133115 IC50 = 1 nM T47101 CM6GV8 137133116 IC50 = 0.8 nM T47101 C5VQU7 137133117 IC50 = 2.8 nM T47101 C4NRV0 137133119 IC50 = 1.8 nM T47101 CTI07K 137133120 IC50 = 2 nM T47101 C45ZQJ 137133121 IC50 = 7.6 nM T47101 CN5AE8 137133122 IC50 = 2.4 nM T47101 CC7P8M 137133125 IC50 = 16.2 nM T47101 CB51RV 137133127 IC50 = 3.6 nM T47101 CM8B9X 137133131 IC50 = 1.2 nM T47101 CL2I8P 137133138 IC50 = 1 nM T47101 CL8QW1 137133139 IC50 = 0.2 nM T47101 CW50HQ 137133141 IC50 = 5.7 nM T47101 CRLW93 137133152 IC50 = 0.6 nM T47101 CU40JZ 137133154 IC50 = 4.1 nM T47101 CJ1ZE9 137133155 IC50 = 1.7 nM T47101 C1W4YT 137205243 IC50 = 6.5 nM T47101 CCM42D 137249694 IC50 > 500 nM T47101 CXC69T 137321158 IC50 = 127 nM T47101 C25ERN 137631967 IC50 = 16.1 nM T47101 CLQT06 137632162 IC50 > 1000 nM T47101 CV49KX 137632804 IC50 > 50000 nM T47101 C0J6IC 137633737 IC50 > 1000 nM T47101 CNX0F9 137634126 IC50 = 10 nM T47101 CI1E8V 137634241 IC50 > 10000 nM T47101 CB35YZ 137634742 IC50 = 456 nM T47101 CMOK58 137634923 IC50 = 3.6 nM T47101 CAW41M 137635785 IC50 = 19200 nM T47101 C5Q1XY 137635805 IC50 = 3.54 nM T47101 CF7P1V 137635991 IC50 > 1000 nM T47101 C2K8LT 137636345 IC50 > 10000 nM T47101 CUR48O 137636669 IC50 = 418.4 nM T47101 CF7O2C 137636828 IC50 > 10000 nM T47101 CPR60M 137637024 IC50 > 10000 nM T47101 C06JRX 137637094 IC50 = 14.5 nM T47101 C6BIO8 137637138 IC50 = 7400 nM T47101 CH2OR6 137637188 IC50 > 1000 nM T47101 CMCI72 137638094 IC50 > 10000 nM T47101 C9R7YH 137638488 IC50 > 20000 nM T47101 C3OVJ8 137638489 IC50 = 4800 nM T47101 C8AI5O 137638529 IC50 = 437.3 nM T47101 CP3SA8 137639345 IC50 > 1000 nM T47101 C7J8FB 137639540 IC50 > 10000 nM T47101 CVBQ91 137640171 IC50 = 12200 nM T47101 CFUX56 137640843 IC50 > 10000 nM T47101 CXM2I8 137640932 IC50 = 10.6 nM T47101 CRQG32 137641135 IC50 = 14.9 nM T47101 C9FH7X 137641558 IC50 = 147.6 nM T47101 C9WBQ0 137641746 IC50 = 127.9 nM T47101 C52EZY 137642247 IC50 = 19999 nM T47101 CGEC59 137642439 IC50 = 6.5 nM T47101 C5E6NQ 137643062 IC50 > 10000 nM T47101 CY8L5M 137644036 IC50 = 591 nM T47101 CJ2M1O 137644088 IC50 = 3.7 nM T47101 C0CTB5 137644554 IC50 > 10000 nM T47101 CS3TU7 137644762 IC50 > 10000 nM T47101 C0P1CJ 137644932 IC50 = 21.1 nM T47101 C9B7XU 137645188 IC50 = 167.3 nM T47101 CK49DP 137645200 IC50 = 8600 nM T47101 CEO3V1 137645361 IC50 > 1000 nM T47101 C58KXF 137645615 IC50 = 19100 nM T47101 CZN04D 137645680 IC50 = 15000 nM T47101 C09CLU 137646239 IC50 > 1000 nM T47101 C79SUZ 137646264 IC50 = 431 nM T47101 C7P5AX 137646321 IC50 > 10000 nM T47101 C0YP8D 137646334 IC50 = 32.3 nM T47101 CSJ4N3 137646379 IC50 = 3300 nM T47101 CBK62Y 137646491 IC50 = 24.9 nM T47101 CZ91YV 137646530 IC50 = 0.7 nM T47101 C7CA9N 137646692 IC50 > 10000 nM T47101 C5IB6V 137647631 IC50 = 14 nM T47101 CS3H8E 137647913 IC50 > 1000 nM T47101 CGF7X2 137647982 IC50 = 200 nM T47101 C1Q8OT 137649334 IC50 = 10000 nM T47101 C7EZP8 137649394 IC50 > 10000 nM T47101 CP2N8Y 137649616 IC50 = 10.4 nM T47101 CBK9F7 137650459 IC50 = 49 nM T47101 CO4HY7 137650511 IC50 = 63.5 nM T47101 C0R2GE 137650566 IC50 = 9300 nM T47101 CHSB74 137650627 IC50 > 10000 nM T47101 CRUE07 137651077 IC50 = 35.2 nM T47101 CI6X0A 137651311 IC50 > 50000 nM T47101 CIM42E 137651341 IC50 > 50000 nM T47101 C1DK0P 137651391 IC50 = 25.2 nM T47101 C47VJA 137651444 IC50 = 91.5 nM T47101 CIR94V 137651828 IC50 > 1000 nM T47101 C6EN8I 137652073 IC50 = 27.9 nM T47101 CU5J4G 137652158 IC50 = 327.4 nM T47101 C0MZ1W 137652333 IC50 = 825.3 nM T47101 CD7UV3 137652920 IC50 = 168.3 nM T47101 CBAF08 137653174 IC50 > 10000 nM T47101 CTV31U 137653424 IC50 > 1000 nM T47101 C6S2ZA 137654098 IC50 = 5.6 nM T47101 C78DVY 137654650 IC50 = 4635 nM T47101 C4B7FC 137655376 IC50 > 1000 nM T47101 CQ85OV 137655810 IC50 > 1000 nM T47101 C86JRT 137656072 IC50 = 11800 nM T47101 C78CUB 137656085 IC50 > 20000 nM T47101 C01JVI 137656138 IC50 = 48.8 nM T47101 CKU8R4 137656214 IC50 = 4800 nM T47101 CFWN28 137657383 IC50 = 219.6 nM T47101 C29AEF 137657653 IC50 = 10800 nM T47101 CWA62P 137657677 IC50 < 4.1 nM T47101 CV5H3Z 137657932 IC50 = 55.8 nM T47101 CSC2G0 137658026 IC50 = 13 nM T47101 C7SEK1 137658232 IC50 > 10000 nM T47101 CQMB10 137658515 IC50 > 50000 nM T47101 CQF74K 137658987 IC50 > 10000 nM T47101 C8DZ6L 137659285 IC50 = 975.1 nM T47101 C4DT3V 137659387 IC50 = 3800 nM T47101 CY8B6K 137659396 IC50 > 1000 nM T47101 CD3K9G 137659884 IC50 > 1000 nM T47101 C9UMG4 137660300 IC50 > 1000 nM T47101 C8D9NE 137660511 IC50 = 2264 nM T47101 CS04UY 137660727 IC50 > 1000 nM T47101 CTJV46 137660921 IC50 = 9500 nM T47101 CIV31M 137661021 IC50 > 1000 nM T47101 CW9U3A 137661140 IC50 > 10000 nM T47101 C82WHL 137661196 IC50 = 66.5 nM T47101 C8WZ2V 137661264 IC50 = 42859 nM T47101 C92NCP 137661343 IC50 = 10000 nM T47101 CK2GY9 137661845 IC50 = 99.3 nM T47101 CK9N2Q 137661928 IC50 = 10400 nM T47101 CM3UF7 137700779 IC50 > 10000 nM T47101 CIWG23 138393067 IC50 = 192 nM T47101 CFR0X3 138454761 IC50 = 31.1 nM T47101 CSRI06 138547901 IC50 = 1.2 nM T47101 C04KQV 138617497 IC50 = 0.6 nM T47101 CUXO19 138617501 IC50 < 0.3 nM T47101 CZ2XH5 139187793 IC50 > 10000 nM T47101 CLRW84 139434103 EC50 = 580 nM T47101 CB6F5R 139434105 EC50 = 890 nM T47101 C7FBY1 139434107 EC50 = 290 nM T47101 CJIH42 139434200 EC50 = 170 nM T47101 C4ID6F 139442949 EC50 = 340 nM T47101 CUH2G6 139554482 IC50 = 4.5 nM T47101 CU0Z1Q 141462232 IC50 = 8.8 nM T47101 CJ2AR3 141462234 IC50 = 1.4 nM T47101 CHP92Q 141462235 IC50 = 0.3 nM T47101 CZH06B 141462237 IC50 = 14 nM T47101 CP1YE3 141462239 IC50 = 0.2 nM T47101 CA7JY9 141462247 IC50 = 0.3 nM T47101 C7C5TV 141462248 IC50 = 3709 nM T47101 C6SQV9 141462249 IC50 = 6.9 nM T47101 CT47AD 141462250 IC50 = 0.2 nM T47101 CC16VK 141462252 IC50 = 10.5 nM T47101 CD38PZ 141462254 IC50 = 14.5 nM T47101 CJ9X4N 141462256 IC50 = 7.2 nM T47101 C6N5HW 141462259 IC50 > 5000 nM T47101 CVR15L 141462267 IC50 = 14.2 nM T47101 CM0UR9 141462270 IC50 = 7.8 nM T47101 C8KSI6 141462272 IC50 = 4.1 nM T47101 CTO7Z2 141462275 IC50 = 74.4 nM T47101 CKG29R 141462277 IC50 = 0.6 nM T47101 C2AMJ0 145351735 IC50 = 10.2 nM T47101 C0DVL8 145351737 IC50 = 12.8 nM T47101 CE7G9J 145351739 IC50 = 1.2 nM T47101 CJN8G2 145351743 IC50 = 6.1 nM T47101 CP67NL 145351755 IC50 = 4.6 nM T47101 CPQ69J 145351756 IC50 = 12.9 nM T47101 C2RUI6 145351760 IC50 = 1.9 nM T47101 CQH4Y8 145351764 IC50 = 2.1 nM T47101 CNC7K1 145351765 IC50 = 1.9 nM T47101 C0ZK6E 145351766 IC50 = 4.1 nM T47101 CNP09Z 145351770 IC50 = 285 nM T47101 CH3I5U 145351773 IC50 = 7.6 nM T47101 C0I6HU 145351778 IC50 > 1000 nM T47101 CKX0Y2 145351783 IC50 = 2 nM T47101 CRV32S 145351784 IC50 = 1.6 nM T47101 CR9W3G 145351797 IC50 = 6.2 nM T47101 C6B3ON 145351798 IC50 = 7.4 nM T47101 CPG63K 145351799 IC50 = 23.5 nM T47101 CO9P7G 145351804 IC50 = 1 nM T47101 C52XUT 145351807 IC50 = 2.8 nM T47101 CY92AL 145351810 IC50 = 3.6 nM T47101 C29XUO 145945978 IC50 = 16.3 nM T47101 CB3Z1W 145949428 IC50 = 200 nM T47101 C15SAP 145949598 IC50 = 9700 nM T47101 CVJS01 145949677 IC50 = 15 nM T47101 CE7H1L 145950269 IC50 = 8800 nM T47101 CL14YA 145950580 IC50 > 100000 nM T47101 CYF32C 145950953 IC50 = 620 nM T47101 CRXJ25 145951211 IC50 = 6600 nM T47101 C1AL5N 145952450 IC50 = 2000 nM T47101 C60XZR 145953297 IC50 = 1800 nM T47101 CAL30B 145953560 IC50 = 140 nM T47101 C0V8SM 145954139 IC50 = 1600 nM T47101 C8VN1Y 145955561 IC50 = 200 nM T47101 CEP8Y7 145955625 IC50 = 36000 nM T47101 C2QOE5 145956264 IC50 = 14000 nM T47101 C1IX5N 145956333 IC50 = 1507 nM T47101 C6ZNJ1 145956488 IC50 = 270 nM T47101 C5VSC7 145956704 IC50 = 167 nM T47101 CB74GR 145957221 IC50 = 4700 nM T47101 C7MBT6 145957742 IC50 = 9900 nM T47101 CB1MI9 145957910 IC50 = 62 nM T47101 CSZ14F 145958261 IC50 = 83000 nM T47101 CS47UF 145958497 IC50 = 94 nM T47101 C1O0QT 145958601 IC50 = 6400 nM T47101 C3V2HG 145960564 IC50 > 500000 nM T47101 C9PKU6 145963750 IC50 = 44 nM T47101 CTUF34 145966712 IC50 = 409 nM T47101 C3Q4XM 145972183 IC50 = 170 nM T47101 CG8R0P 145972697 IC50 = 61 nM T47101 C2QL9C 145980124 IC50 > 1000 nM T47101 C93AOR 145980752 IC50 = 280 nM T47101 CFCD85 145981675 IC50 = 8.2 nM T47101 C03PYD 145986466 IC50 < 1000 nM T47101 CX5CD2 145987573 IC50 > 1000 nM T47101 CVG9P7 145987920 IC50 = 22.2 nM T47101 CRC4D9 145988151 IC50 = 1.2 nM T47101 C5VLI4 145988744 IC50 = 67.5 nM T47101 C9DJM6 145990718 IC50 = 132 nM T47101 CZMK39 145990966 IC50 = 36.1 nM T47101 CUHW41 145991304 IC50 > 1000 nM T47101 CS7TD1 145993995 IC50 > 10000 nM T47101 CN7EF3 145996526 IC50 > 1000 nM T47101 CBM7C5 146773032 IC50 = 16230 nM T47101 C9D1EH 147117461 IC50 = 21560 nM T47101 C8I1HV 147384518 IC50 = 26470 nM T47101 C7DYK4 147709549 IC50 = 28150 nM T47101 CIT79C 148291912 IC50 = 16250 nM T47101 C2U0SJ 148390225 IC50 = 36980 nM T47101 CJ23ZE 148637488 IC50 = 18220 nM T47101 CVL49H 149513019 IC50 = 33450 nM T47101 CR20QN 149611945 IC50 = 808 nM T47101 CSE96B 152685456 IC50 = 1103 nM T47101 CFKU39 152790957 IC50 = 58940 nM T47101 CV41DF 153011787 IC50 = 35890 nM T47101 CC2AQ0 154573782 IC50 = 8340 nM T47101 COZA72 155415442 IC50 = 12 nM T47101 C82YKF 155415443 IC50 > 10000 nM T47101 CQC20K 155415472 IC50 = 373 nM T47101 CL98BI 155415495 IC50 = 119 nM T47101 C4GZ7D 155415496 IC50 = 1050 nM T47101 C8UOT3 155415499 IC50 = 17 nM T47101 CHKX30 155415500 IC50 > 10000 nM T47101 C94HAT 155415504 IC50 = 391 nM T47101 CYD73X 155415508 IC50 > 3330 nM T47101 CMJZ23 155415509 IC50 = 72 nM T47101 C09YSN 155415512 IC50 = 89 nM T47101 CNF0X5 155415516 IC50 > 10000 nM T47101 CJ0DO6 155415524 IC50 > 10000 nM T47101 CK8Y9I 155415561 IC50 > 10000 nM T47101 C59VKN 155415568 IC50 = 20 nM T47101 CGM4U0 155415583 IC50 = 6710 nM T47101 CS0Y1T 155512636 IC50 = 10.1 nM T47101 C9X8LP 155513025 IC50 = 1.7 nM T47101 C2MD1Q 155513187 IC50 > 10000 nM T47101 CU12GD 155513666 IC50 = 18520 nM T47101 CL75PC 155515231 IC50 > 10000 nM T47101 CU76NE 155516227 IC50 = 47520 nM T47101 C86HPW 155518524 IC50 = 13000 nM T47101 C2HL6O 155519199 IC50 > 10000 nM T47101 CL3DV0 155519320 IC50 = 0.4 nM T47101 C8S1YX 155519682 IC50 = 16.5 nM T47101 C9HEY1 155519702 IC50 = 45260 nM T47101 CU6Z5O 155520650 IC50 = 130 nM T47101 C7FIU3 155520706 IC50 = 12.9 nM T47101 C1ID9A 155523715 IC50 = 55.4 nM T47101 CY6NE1 155523855 IC50 = 230 nM T47101 C1DY8F 155524432 IC50 = 25.4 nM T47101 CRP7Q6 155525519 IC50 = 300 nM T47101 CS1U2Z 155526433 IC50 = 26.8 nM T47101 CHD8E5 155527081 IC50 = 6.7 nM T47101 CFUG34 155527917 IC50 = 11.7 nM T47101 CTD5R7 155528337 IC50 = 310 nM T47101 C9P2NQ 155528441 IC50 = 17230 nM T47101 CLEJ03 155529517 IC50 = 380 nM T47101 CFRQ41 155530069 IC50 = 2.4 nM T47101 CHSA34 155530353 IC50 = 8.8 nM T47101 CFB02G 155532218 IC50 = 20.7 nM T47101 C3NZO0 155533789 IC50 = 460 nM T47101 C2DJ0A 155534253 IC50 = 390 nM T47101 C37RFQ 155534994 IC50 = 480 nM T47101 CD8TO7 155535214 IC50 = 25450 nM T47101 C3LC9I 155536820 IC50 = 961.7 nM T47101 CX37HC 155537699 IC50 > 1000 nM T47101 CI26FR 155538679 IC50 = 6.4 nM T47101 C1VJH0 155543634 IC50 = 62150 nM T47101 CW4FU3 155546952 IC50 > 100 nM T47101 C0BRU3 155547256 IC50 > 10000 nM T47101 C3S8MD 155547644 IC50 = 42.4 nM T47101 C5SXH4 155547874 IC50 = 6.7 nM T47101 CE6M4K 155548572 IC50 = 1217 nM T47101 CD8A5R 155549158 IC50 = 19.3 nM T47101 C6URZ7 155550475 IC50 = 390 nM T47101 C9WN5D 155554550 IC50 = 0.9 nM T47101 CUA73V 155555832 IC50 = 170 nM T47101 CWDR07 155555935 IC50 = 22160 nM T47101 CFC8B0 155557936 IC50 = 11.5 nM T47101 CX06SK 155558020 IC50 = 3.9 nM T47101 C8L6PM 155561965 IC50 = 610 nM T47101 C2L5MS 155563171 IC50 = 11.6 nM T47101 C81JZW 155563388 IC50 = 280 nM T47101 C21DWP 155564268 IC50 = 2 nM T47101 CAU45D 155565428 IC50 = 3.2 nM T47101 CM23DI 155565660 IC50 = 420 nM T47101 C3MK6Z 155567552 IC50 = 9 nM T47101 CF1W4I 155568065 IC50 = 20.1 nM T47101 CK10HA 155568167 IC50 = 280 nM T47101 CIN82D 155568305 IC50 = 389.3 nM T47101 C94IJB 10367131 IC50 = 7 nM T47101 C13GYL 127031746 IC50 < 5000 nM T47101 CI8LX0 57976125 IC50 = 8 nM T47101 D00ERW 44444843 Ki > 4737 nM T47101 D00GVV 5329155 IC50 = 13300 nM T47101 D00TBD 10461815 IC50 = 3000 nM T47101 D00YCU 667662 IC50 = 6400 nM T47101 D01FWD 606669 IC50 > 50000 nM T47101 D01MUN 5328453 IC50 > 50000 nM T47101 D02BXJ 46864270 IC50 = 1.8 nM T47101 D02XKJ 5328466 IC50 = 22000 nM T47101 D03DZO 11715767 IC50 > 10000 nM T47101 D03NPX 447077 IC50 = 1250 nM T47101 D04FNY 25195216 IC50 = 100 nM T47101 D04ZWF 53396311 IC50 > 1000 nM T47101 D06FFZ 91827382 IC50 = 2.9 nM T47101 D06HVH 54613583 IC50 > 10000 nM T47101 D06QUJ 24180722 IC50 = 1900 nM T47101 D07IHM 9823787 IC50 > 10000 nM T47101 D07OSK 6419834 IC50 = 5000 nM T47101 D08HFG 24809764 IC50 > 10000 nM T47101 D08RZB 11153014 IC50 > 10000 nM T47101 D09HVH 135566652 IC50 > 10 nM T47101 D09LPL 5329103 IC50 = 170 nM T47101 D09QBA 23378546 IC50 > 10000 nM T47101 D0A4XJ 5289418 IC50 = 30 nM T47101 D0C2GE 67161540 IC50 = 6 nM T47101 D0C6KI 5329006 IC50 = 7000 nM T47101 D0D5EW 5311104 IC50 = 934 nM T47101 D0E7VO 59627005 IC50 = 8.7 nM T47101 D0EE6A 6398883 IC50 > 10000 nM T47101 D0GW4Q 5330524 IC50 = 933 nM T47101 D0HE0E 5941540 IC50 = 10000 nM T47101 D0K2YG 5328512 IC50 = 18000 nM T47101 D0KH5T 5687 IC50 = 11000 nM T47101 D0O6OH 71553154 IC50 = 1710 nM T47101 D0OH3J 5330526 IC50 = 244 nM T47101 D0P3JW 447700 IC50 = 61.5 nM T47101 D0P6JS 11675054 IC50 > 10000 nM T47101 D0Q3KS 9957049 IC50 > 5000 nM T47101 D0R2WK 16038120 IC50 = 19 nM T47101 D0S1KJ 5328733 IC50 = 100 nM T47101 D0T8NU 16757525 IC50 > 4000 nM T47101 D0US9O 45275255 IC50 = 50 nM T47101 D0XC6G 135464491 IC50 = 1400 nM T47101 D0XS9E 5330535 IC50 > 10000 nM T47101 D0YE1X 9927943 IC50 > 100000 nM T47101 D0YZ7H 9797370 IC50 = 45800 nM T47101 D0Z7GH 5330525 IC50 = 451 nM T47101 D0Z7TM 22273644 IC50 = 78 nM T00407 D08HVE 679 IC50 = 280000000 nM T00407 D0E3SH 6918837 IC50 = 5 nM T00407 D0E7PQ 5311 IC50 = 10 nM T00407 D0L7LC 5352062 IC50 = 36 nM T00407 D00BYM 10461508 IC50 = 1070 nM T00407 D01LVE 57389999 IC50 = 39 nM T00407 D02YNI 9936746 Ki = 5.7 nM T00407 D03NJY 66577114 IC50 = 5300 nM T00407 D05ICT 132010322 Ki = 1.6 nM T00407 D06QBV 90647162 IC50 = 8 nM T00407 D07OFM 46943432 Ki = 23 nM T00407 D0G8BM 16722836 IC50 = 290 nM T00407 D0M2TS 71600087 IC50 = 1 nM T00407 D0O0LQ 11364421 IC50 = 25 nM T00407 D0PH9I 118693659 Ki = 5 nM T00407 D0XT6W 6918638 IC50 = 27 nM T00407 D0ZW4W 46907787 Ki = 5.3 nM T00407 D09FVR 122553422 IC50 < 11 nM T00407 D0HB3F 118340554 Ki < 1 nM T00407 D0KG9M 19910 IC50 = 980 nM T00407 D0SG9F 86566737 IC50 = 10 nM T00407 D09SFV 3973 IC50 = 12400 nM T00407 D0D3PX 46926350 IC50 = 19000 nM T00407 CL80QG 11820 IC50 = 73000 nM T00407 CZI4N9 13387 IC50 = 2660000 nM T00407 C5XSG3 19868 IC50 = 220000 nM T00407 C2BW3V 97075 IC50 = 34200 nM T00407 C4ZJO2 108402 IC50 = 6880000 nM T00407 CX0Z2S 205810 IC50 > 10000 nM T00407 CVG54O 209396 IC50 > 10000 nM T00407 CZX1K3 223771 IC50 > 200000 nM T00407 CD8OI6 251290 IC50 = 125892.54 nM T00407 C2IJU0 440987 IC50 = 39810.72 nM T00407 CJ6X2Y 572983 IC50 = 80000 nM T00407 CS7Z2U 584972 IC50 = 2870 nM T00407 CAT79Z 589098 IC50 > 100000 nM T00407 CPUC56 594190 IC50 = 101 nM T00407 CG5O0H 638578 IC50 = 18400 nM T00407 CG8C3X 651118 IC50 = 13300 nM T00407 C3CO8M 699832 IC50 = 210 nM T00407 CB3M7R 701320 IC50 = 47280 nM T00407 CB7ZY9 714750 IC50 = 5770 nM T00407 C4QD1V 723220 IC50 > 10000 nM T00407 CM1EX8 735746 IC50 = 3700000 nM T00407 COP70H 735747 IC50 = 260000 nM T00407 C4HEN5 739455 IC50 = 1000 nM T00407 CT41GY 747882 IC50 > 30000 nM T00407 CLN68U 750666 IC50 = 11000 nM T00407 CRN2X9 781532 IC50 = 47280 nM T00407 CX5U7E 781533 IC50 = 1910 nM T00407 CM71KW 786866 IC50 = 3000 nM T00407 CLC4D8 827656 IC50 > 10000 nM T00407 CT2J6Y 845994 IC50 = 27520 nM T00407 CB1Q6P 872951 IC50 = 71000 nM T00407 CV6DC3 878890 IC50 = 337 nM T00407 CS9GR8 893324 IC50 = 23060 nM T00407 CR65HV 975948 IC50 = 18720 nM T00407 C29JXM 984803 IC50 = 3020 nM T00407 C3UW5D 986642 IC50 > 10000 nM T00407 CQEF34 1002773 IC50 > 100000 nM T00407 CZ60SO 1015929 IC50 = 5730 nM T00407 CT48GV 1069056 IC50 = 530 nM T00407 C50QOJ 1069081 IC50 = 2280 nM T00407 CBG2A0 1078352 IC50 > 20000 nM T00407 CZP8B2 1090309 IC50 = 4800 nM T00407 CFA3Q8 1090310 IC50 = 4800 nM T00407 CV2ES8 1192817 IC50 = 130 nM T00407 CD0S4T 1220046 IC50 = 50750 nM T00407 C5TSY1 1244585 IC50 = 15530 nM T00407 CHP0C9 1380882 IC50 = 18000 nM T00407 CF3XV1 1382046 IC50 = 20000 nM T00407 C0TSA6 1395662 IC50 = 237.4 nM T00407 C92EYR 1503595 IC50 = 30000 nM T00407 CRT85V 1511056 IC50 = 69230 nM T00407 C2M0SE 1511198 IC50 = 1995.26 nM T00407 CJK1F0 1511199 IC50 = 1258.93 nM T00407 CZG1R8 1523399 IC50 = 3240 nM T00407 CI7UJ2 1523400 IC50 = 3740 nM T00407 C0A2LP 1523407 IC50 = 9680 nM T00407 C83WZI 1523409 IC50 = 4700 nM T00407 CY42VE 1534872 IC50 = 1530 nM T00407 CF1GQ2 1535153 IC50 = 1000 nM T00407 C7XRT1 1581020 IC50 = 1550 nM T00407 CCNQ31 1585889 IC50 = 1110 nM T00407 CP1L8I 1652717 IC50 = 1040 nM T00407 C31ITR 1895574 IC50 = 2100 nM T00407 CUVQ31 1922908 IC50 = 6600 nM T00407 CCJL62 2317823 IC50 > 10000 nM T00407 CP5GB0 2347699 IC50 = 769.2 nM T00407 C4T2JC 2371015 IC50 = 8940 nM T00407 C4Q0LV 2673048 IC50 > 100000 nM T00407 COZK67 2728636 IC50 = 43000 nM T00407 CDRT80 2782959 IC50 = 80900 nM T00407 CH95GA 2787707 IC50 = 8500 nM T00407 CHOL56 2824992 IC50 = 7500 nM T00407 C9V8HM 2841849 IC50 = 2100 nM T00407 C0EN8Y 2854307 IC50 > 10000 nM T00407 C8MB5Z 2874948 IC50 = 10980 nM T00407 C2OHC6 2927305 IC50 = 23000 nM T00407 C3DT1H 2973846 IC50 = 42230 nM T00407 CV9W7S 2988057 IC50 = 15800 nM T00407 C9PS6J 3109203 IC50 > 10000 nM T00407 CA89QB 3113698 IC50 = 370 nM T00407 C9RJG0 3132761 IC50 = 5360 nM T00407 CXD3U8 3152392 IC50 > 200000 nM T00407 CCS0Y2 3156673 IC50 = 738 nM T00407 CT1RG9 3293096 IC50 = 32230 nM T00407 C8GXW4 3319300 IC50 > 100000 nM T00407 CM1AE9 3370466 IC50 > 50118.72 nM T00407 CIE1C5 3499770 IC50 = 3400 nM T00407 CGE54P 3573716 IC50 > 50118.72 nM T00407 CS9M8A 3577407 IC50 > 50118.72 nM T00407 CJ4U6Y 3589423 IC50 = 5011.87 nM T00407 C2U9DI 3657707 IC50 = 39810.72 nM T00407 CPN2V4 3673391 IC50 > 50118.72 nM T00407 CYOV56 3681703 IC50 = 12589.25 nM T00407 C1KHJ6 3692581 IC50 = 3090 nM T00407 CB2ZP4 3721448 IC50 = 10940 nM T00407 C2P6IC 3846558 IC50 = 39000 nM T00407 C6KDA4 3900479 IC50 = 2103 nM T00407 CMDG67 3964313 IC50 = 50920 nM T00407 C42AQR 4102773 IC50 > 14000 nM T00407 C28EBX 4790771 IC50 = 39810.72 nM T00407 CY71BJ 4800411 Ki = 350 nM T00407 CR3SF5 4907545 IC50 = 5011.87 nM T00407 CWG19Q 4908238 IC50 = 19952.62 nM T00407 CB1HV6 4912924 IC50 > 100000 nM T00407 CXBG75 5125956 IC50 > 501187.23 nM T00407 C8BZ9Y 5325760 IC50 = 65000 nM T00407 CT8G2Z 6458480 IC50 > 50118.72 nM T00407 CEAN08 6611008 IC50 = 300 nM T00407 CLVK27 7731152 IC50 > 30000 nM T00407 C81TXG 8781434 IC50 = 2010 nM T00407 C5K3IF 9404764 IC50 = 34500 nM T00407 CC7IO0 9497211 IC50 = 890 nM T00407 C93EDN 10442296 IC50 > 100000 nM T00407 C5Y1WP 11128828 IC50 = 7000 nM T00407 C0BW3Q 11260691 IC50 = 84 nM T00407 CMJ01U 11283298 IC50 = 109 nM T00407 C6ALO2 11511524 Ki = 60 nM T00407 CE5K4J 11577250 IC50 = 25 nM T00407 CT53WA 12206142 IC50 > 200000 nM T00407 C1C6KY 12478742 Ki = 12000 nM T00407 C4H9EO 12488974 Ki = 21000 nM T00407 C34GWI 12622087 IC50 = 60000 nM T00407 CIG94A 13953713 IC50 = 19952.62 nM T00407 CTB86M 14774292 IC50 = 51000 nM T00407 CWPN42 15052068 IC50 = 12710 nM T00407 CQS67F 15944463 IC50 = 1090 nM T00407 CI82RX 15944465 IC50 > 30000 nM T00407 CP3EN5 15944506 IC50 = 1960 nM T00407 CP85DF 15944510 IC50 = 6490 nM T00407 CO8J4E 15944522 IC50 = 8220 nM T00407 C4E0UM 15944523 IC50 = 440 nM T00407 CTLV13 15944527 IC50 = 310 nM T00407 CN08ZF 15944528 IC50 = 9570 nM T00407 C1KAE2 15978962 IC50 = 33.9 nM T00407 CO3IL6 15990226 IC50 > 50118.72 nM T00407 CZ91JF 15990296 IC50 > 50118.72 nM T00407 C9K1AY 16228516 IC50 = 670 nM T00407 CCF3G5 16232084 IC50 > 50000 nM T00407 C1W7TE 16258532 IC50 = 10000 nM T00407 CP60ON 16258758 Ki = 1200 nM T00407 CE3X0C 16265714 Ki = 370 nM T00407 C25EUG 16272810 IC50 > 50118.72 nM T00407 CK2ES3 16313990 IC50 > 50118.72 nM T00407 CZ59FR 16316459 IC50 > 50118.72 nM T00407 CEN83U 16323492 IC50 > 50118.72 nM T00407 CM1R8O 16344932 IC50 = 31622.78 nM T00407 CQ3A6K 16371566 IC50 = 7400 nM T00407 CO6HM1 16480179 IC50 = 26000 nM T00407 CC17UZ 16654419 IC50 = 21270 nM T00407 CT5N9A 16654554 IC50 = 13850 nM T00407 CNK13T 16654568 IC50 = 11180 nM T00407 C4TC3X 16722832 IC50 = 130 nM T00407 CKJB19 16728035 IC50 = 18610 nM T00407 CY10PK 16728036 IC50 = 1640 nM T00407 CGFA68 16822024 Ki = 300 nM T00407 CO8M7K 17405877 IC50 = 199526.23 nM T00407 CIN8H3 17443248 IC50 = 19530 nM T00407 C9IP3Q 17446910 IC50 > 50118.72 nM T00407 CM09CN 17481591 IC50 = 24000 nM T00407 CLQ34F 17488246 IC50 = 160030 nM T00407 CO6KM2 17498966 IC50 > 100000 nM T00407 CVGU58 18536615 IC50 = 2900 nM T00407 CI8Z3Q 18536630 IC50 = 2500 nM T00407 C6Y4GF 18536633 IC50 = 3700 nM T00407 CDS15V 18536647 IC50 = 24000 nM T00407 C0DWP2 19596259 IC50 = 1810 nM T00407 CP7M5X 19704956 IC50 = 100 nM T00407 C4I2NX 20946734 IC50 > 50118.72 nM T00407 CDF52J 21680034 IC50 = 30000 nM T00407 C9IZ8A 21914263 IC50 = 4110000 nM T00407 C12TZA 22432992 IC50 > 50118.72 nM T00407 CXL15A 22433053 IC50 > 50118.72 nM T00407 CU9A5T 22696534 IC50 > 30000 nM T00407 C51GQD 24043179 Ki = 160000 nM T00407 CW5HI1 24156462 IC50 = 820 nM T00407 CLP9S1 24687782 IC50 > 50118.72 nM T00407 CIBE92 24789797 IC50 > 50118.72 nM T00407 COB70I 24789844 IC50 > 50118.72 nM T00407 C2JIY3 24790912 IC50 > 50118.72 nM T00407 C4S6OT 24906340 IC50 > 30000 nM T00407 CX2Q9M 24906350 IC50 = 6930 nM T00407 C49GBY 27604952 IC50 = 74000 nM T00407 CZ0JV1 27770210 IC50 = 6400 nM T00407 CN0J2C 29180108 IC50 > 50118.72 nM T00407 CAE73B 30342829 IC50 = 8180 nM T00407 C9OMZ0 30342838 IC50 = 3650 nM T00407 CQBK46 30342991 IC50 = 2050 nM T00407 CV6PQ8 30342999 IC50 = 810 nM T00407 CMQX14 30343069 IC50 = 4560 nM T00407 CI4AQ1 39129690 IC50 = 42000 nM T00407 C3UFS6 39791103 IC50 = 4800 nM T00407 C1OEL5 40889550 IC50 = 5200 nM T00407 CMN7L1 43286729 IC50 = 24000 nM T00407 C7KG1R 43286787 IC50 > 100000 nM T00407 C2P0IW 44243549 IC50 = 24600 nM T00407 C1C3QM 44269241 IC50 > 250000 nM T00407 C3VRO9 44557921 IC50 > 10000 nM T00407 C0GIA6 45103903 IC50 > 10000 nM T00407 CK3NP1 46249107 IC50 > 50118.72 nM T00407 C5HXW9 46249116 IC50 > 50118.72 nM T00407 CD06LA 46249215 IC50 = 10000 nM T00407 CCE1S0 47026724 IC50 = 27000 nM T00407 C3EL4J 47083668 IC50 = 8810 nM T00407 CT48OH 47108307 IC50 > 10000 nM T00407 C5FMU9 49169334 IC50 = 60000 nM T00407 C8H4PR 49766616 IC50 = 39040 nM T00407 CR87KB 49805721 Ki = 199.53 nM T00407 CN67BI 49805848 Ki = 398.11 nM T00407 C98BLM 49871817 IC50 = 26 nM T00407 C60BPW 49871818 IC50 > 10000000 nM T00407 CXC9K3 51003468 IC50 = 398.11 nM T00407 CI50XM 51063711 IC50 = 1700 nM T00407 C35MQH 51371083 IC50 > 20000 nM T00407 CTFL63 52100397 IC50 = 42230 nM T00407 CPSE59 52106219 IC50 = 10980 nM T00407 CWQ5G6 52106229 IC50 = 21130 nM T00407 CN5XV2 52106240 IC50 = 5210 nM T00407 C1PBE9 52233794 IC50 = 4630 nM T00407 C24YBT 52233800 IC50 = 11870 nM T00407 CHD35F 52233804 IC50 = 3340 nM T00407 CE4XV7 52233933 IC50 = 6540 nM T00407 CG3PR6 52912222 IC50 = 0.3981 nM T00407 CI68XL 52912223 IC50 = 280 nM T00407 CBXV52 52932793 IC50 = 251.19 nM T00407 CJE59U 52932930 IC50 = 1584.89 nM T00407 CSZ2T6 52932933 IC50 = 3162.28 nM T00407 CN87IR 52933159 IC50 = 794.33 nM T00407 CG6OL4 52933160 IC50 = 501.19 nM T00407 CP8Y9K 52933161 IC50 = 1258.93 nM T00407 CK8Z4P 52933165 IC50 = 3981.07 nM T00407 CKC17F 52933403 IC50 = 1258.93 nM T00407 CD08ZX 52933405 IC50 = 1000 nM T00407 C1T7VQ 52933407 IC50 = 1584.89 nM T00407 CE65VO 52933414 IC50 = 501.19 nM T00407 CFS84O 52933416 IC50 = 501.19 nM T00407 CO8VX9 52933655 IC50 = 1258.93 nM T00407 C6G7BE 52933893 IC50 = 794.33 nM T00407 C7VN1E 52934039 IC50 = 1000 nM T00407 CUZE18 52934122 IC50 = 501.19 nM T00407 CN16FE 52934128 IC50 = 6309.57 nM T00407 CTS13B 52934275 IC50 = 3981.07 nM T00407 CX3BI9 52934358 IC50 = 1995.26 nM T00407 CNOH36 52935183 IC50 = 251.19 nM T00407 CLRH53 52935478 IC50 = 1258.93 nM T00407 C53EFC 52935914 IC50 = 398.11 nM T00407 CXP76N 52936135 IC50 = 251.19 nM T00407 CJIB35 53054190 IC50 = 6000 nM T00407 C6V8YR 53054191 IC50 = 16000 nM T00407 C09HTR 53054200 IC50 = 1200 nM T00407 CUS8F7 53054236 IC50 = 7600 nM T00407 CX5QN4 53054237 IC50 = 20000 nM T00407 CD2TY9 53054238 IC50 = 11000 nM T00407 C47GAW 53054240 IC50 = 8200 nM T00407 CVH2G1 53054241 IC50 = 5600 nM T00407 CF9E2V 53054248 IC50 = 2600 nM T00407 CRWK92 53054249 IC50 = 5600 nM T00407 CSXI51 53054250 IC50 = 2000 nM T00407 CM12EL 53054251 IC50 = 3300 nM T00407 CY5L3J 53054252 IC50 = 4500 nM T00407 CWV76Y 53054258 IC50 = 1100 nM T00407 CIU8P7 53054259 IC50 = 500 nM T00407 CVX3R0 53054274 IC50 = 3300 nM T00407 CB05OM 53054276 IC50 = 1800 nM T00407 CLR97U 53054289 IC50 = 1000 nM T00407 CJ6E2Q 53054291 IC50 = 4400 nM T00407 C1WSZ4 53054297 IC50 = 2400 nM T00407 C7A2XC 53054319 IC50 = 3000 nM T00407 C0J1EO 53054320 IC50 = 6600 nM T00407 CK68UF 53054321 IC50 = 1200 nM T00407 CJY5S2 53054322 IC50 = 4200 nM T00407 C1YW5L 53054324 IC50 = 2800 nM T00407 C8Q6WG 53054325 IC50 = 1800 nM T00407 CJHR65 53268658 IC50 > 10000 nM T00407 CH6I4T 53268667 IC50 > 10000 nM T00407 CRG95D 53268718 IC50 = 1020 nM T00407 CQEF28 53308655 IC50 = 51200 nM T00407 C9V5LX 53318989 IC50 = 15.5 nM T00407 C7WVX3 54695746 IC50 = 2830 nM T00407 CEK3X6 54757749 IC50 = 23200 nM T00407 C1D3WH 54757750 IC50 = 9700 nM T00407 C1DZ7Y 54757751 IC50 = 7700 nM T00407 C6W5OZ 54757752 IC50 = 7500 nM T00407 C1KWY4 54759170 IC50 = 10000 nM T00407 CM8Y7O 56697168 IC50 = 13260 nM T00407 C7HK2C 56924692 IC50 = 2600 nM T00407 CTVM34 56929801 IC50 = 380.19 nM T00407 CX6SD9 56950289 IC50 = 3200 nM T00407 CZ6NE0 56950420 IC50 = 2500 nM T00407 CJ5BE9 56950421 IC50 = 5200 nM T00407 CL96VQ 56950422 IC50 = 3000 nM T00407 CCLD98 56950423 IC50 = 13000 nM T00407 CZD7G2 56950424 IC50 = 6500 nM T00407 CPQ0B7 56950425 IC50 = 7400 nM T00407 CL90DK 56950426 IC50 = 1000 nM T00407 CF9IJ1 56950561 IC50 = 1300 nM T00407 CH24QC 56950562 IC50 = 12000 nM T00407 CU62NO 56950563 IC50 = 17000 nM T00407 CRD86M 56950564 IC50 = 15000 nM T00407 CNQ2L5 56950565 IC50 = 22000 nM T00407 CB3A1Z 56950566 IC50 = 10000 nM T00407 C5ADP4 56950567 IC50 = 17000 nM T00407 CFW0D1 57339435 IC50 = 1258.93 nM T00407 C56SWR 57344430 IC50 = 6200 nM T00407 C3ZXF4 57344431 IC50 = 36 nM T00407 CU74JQ 57344432 IC50 = 1100 nM T00407 CEK82U 57344527 IC50 = 2200 nM T00407 CE71PA 57344528 IC50 = 86 nM T00407 C6OZU2 57344531 IC50 = 200 nM T00407 CE37LA 57344606 IC50 = 190 nM T00407 CEP6Q1 57345408 IC50 < 500 nM T00407 CCU1P9 57388845 IC50 = 5700 nM T00407 C0Z9HP 57389114 IC50 = 2100 nM T00407 C31KUT 59149763 Ki = 251.19 nM T00407 CF8B4E 60498769 IC50 = 5000 nM T00407 CYL1B0 66553124 IC50 = 1900 nM T00407 CKC51O 66553125 IC50 = 4800 nM T00407 CW8K1P 67173666 IC50 = 7943.28 nM T00407 CPD6G3 67192581 IC50 = 1258.93 nM T00407 CX17NA 67195278 IC50 = 501.19 nM T00407 CPY59D 67195867 IC50 = 25118.86 nM T00407 C0QK5F 67814495 IC50 = 250 nM T00407 CN3KZ8 68161075 IC50 = 398.11 nM T00407 C49IOA 68161669 IC50 = 501.19 nM T00407 CJ7N3M 68184870 IC50 = 1258.93 nM T00407 CT4Z2A 68184871 IC50 = 501.19 nM T00407 CEX74I 68186034 IC50 = 5011.87 nM T00407 CCE3I0 68199877 IC50 = 33 nM T00407 C25INY 68204735 IC50 = 1258.93 nM T00407 C6KWC8 69236418 IC50 > 200000 nM T00407 CMC7V5 70664240 IC50 = 1258.93 nM T00407 CDY89S 70680609 IC50 > 50000 nM T00407 C1I6OH 70681167 IC50 = 7943.28 nM T00407 C7GJW9 70681170 IC50 = 630.96 nM T00407 C8H4JX 70681173 IC50 = 794.33 nM T00407 C6NYK2 70681174 IC50 = 501.19 nM T00407 C8KBJ0 70683271 IC50 = 1258.93 nM T00407 CXD3F9 70691699 IC50 = 398.11 nM T00407 C9L0KD 70699440 IC50 = 386 nM T00407 CV7OR2 70699441 IC50 = 380.19 nM T00407 C76BEK 71271375 IC50 = 390 nM T00407 C0HTY9 71271805 IC50 = 880 nM T00407 CJ90CI 71271897 IC50 = 220 nM T00407 C76ZPW 71271926 IC50 = 600 nM T00407 CR96WH 71271969 IC50 = 4400 nM T00407 C2P4GJ 71272064 IC50 = 360 nM T00407 C5YBX2 71272103 IC50 = 730 nM T00407 C7VJK4 71272293 IC50 = 180 nM T00407 C1UZ4Q 71272605 IC50 = 2300 nM T00407 CFSP50 71297183 IC50 = 790 nM T00407 COZ1E0 71297184 IC50 = 4100 nM T00407 CB2NY9 71297185 IC50 = 4100 nM T00407 CS1BL2 71450122 IC50 = 880 nM T00407 CL8Y9N 71450297 IC50 = 1258.93 nM T00407 CUY20J 71459124 IC50 = 470 nM T00407 C6CQT5 71462842 IC50 = 6309.57 nM T00407 CWUE65 71532084 IC50 = 27 nM T00407 CMJC68 71615940 Ki = 3.1 nM T00407 CONT42 71615943 Ki = 6.4 nM T00407 C6U5KC 71615944 Ki = 4.1 nM T00407 CTXM79 71616053 Ki = 1.5 nM T00407 C2U7NS 71616054 Ki = 2.9 nM T00407 CLZ7X1 71616055 Ki = 14 nM T00407 CXLN73 71616297 Ki = 48 nM T00407 C7UQH0 71616300 Ki = 2.4 nM T00407 C47LAI 71616301 Ki = 4.4 nM T00407 CR3M1X 71616302 Ki = 9.8 nM T00407 C93NFZ 71616418 Ki = 32 nM T00407 CN1H9P 71616658 Ki = 4.5 nM T00407 CY20JZ 71616659 Ki = 68 nM T00407 C25ZDV 71616989 Ki = 3.6 nM T00407 C82EAI 71617108 Ki = 9.4 nM T00407 C1UA6X 71617219 Ki = 5.8 nM T00407 C4O7ZL 71617338 Ki = 68 nM T00407 C1SHR7 71617458 Ki = 12 nM T00407 CYI2A3 71617461 Ki = 19 nM T00407 CE91KU 71617462 Ki = 3.7 nM T00407 C7BU8M 71621544 Ki = 6.3 nM T00407 C4MJ0T 71624784 IC50 = 640 nM T00407 CIX91F 71624785 IC50 = 1700 nM T00407 C1D8GF 71624786 IC50 = 1500 nM T00407 C3R9WA 71624787 IC50 = 3900 nM T00407 CLQ1X8 71624896 IC50 = 2600 nM T00407 COW9G4 71624897 IC50 = 544 nM T00407 CODK30 71624901 IC50 = 1360 nM T00407 CI15JC 71624902 IC50 = 1380 nM T00407 CLZ7C8 71624903 IC50 = 1170 nM T00407 CLA71B 71661332 IC50 = 3700 nM T00407 CW5F3S 71661333 IC50 = 10000 nM T00407 C7US6G 71661335 IC50 = 22800 nM T00407 CP0C3Q 71661522 IC50 = 23800 nM T00407 C13DUN 71661524 IC50 = 3300 nM T00407 C9WZO5 71661707 IC50 = 3500 nM T00407 C7FW1U 71661708 IC50 = 2600 nM T00407 CG3U8D 71661709 IC50 = 2400 nM T00407 CAYC45 71661710 IC50 = 2500 nM T00407 C0TK5C 71661712 IC50 = 230 nM T00407 C1FD9C 71661885 IC50 = 2200 nM T00407 C74UGA 71661886 IC50 = 570 nM T00407 C1VXA5 71664045 IC50 = 50700 nM T00407 CWJR48 71664046 IC50 = 2600 nM T00407 C7GY3D 71664047 IC50 = 4400 nM T00407 CX8B7F 71717163 IC50 = 58.7 nM T00407 CG10TU 71720056 IC50 = 180 nM T00407 CS26GP 71747837 IC50 > 10000 nM T00407 CIPN50 71760902 Ki = 15 nM T00407 C74CSP 71811952 EC50 = 7100 nM T00407 CMZU93 71811973 EC50 = 280 nM T00407 CZQ4G1 71812037 EC50 = 75 nM T00407 CHDB19 71812048 Ki = 210 nM T00407 CA1F7L 71812065 Ki = 91 nM T00407 C1IHP6 71812067 Ki = 250 nM T00407 CX73WV 71862498 IC50 = 63280 nM T00407 CD1FE6 71935082 IC50 = 1900 nM T00407 CIYP36 71938587 IC50 = 3000 nM T00407 CL0NM3 71942353 IC50 = 24000 nM T00407 C7FVU5 71970469 IC50 = 11720 nM T00407 C1OGC5 71975056 IC50 = 21000 nM T00407 CGP24T 72201024 IC50 = 2511.89 nM T00407 CA81BL 72201025 IC50 = 4100 nM T00407 CA71SN 72203613 IC50 = 14 nM T00407 C9M6QY 72547793 Ki = 2.6 nM T00407 CTQ9S3 72548029 Ki = 5.6 nM T00407 CUI57F 72548032 Ki = 17 nM T00407 CW4QJ6 72548735 Ki = 14 nM T00407 C4L6PB 72549215 Ki = 140 nM T00407 C01LXD 72549905 Ki = 58 nM T00407 C64NRP 72550116 Ki = 13 nM T00407 C4VBJ1 72684073 IC50 = 1258.93 nM T00407 C2AFW1 72702849 IC50 = 398.11 nM T00407 C3R1IL 72703043 IC50 = 100000 nM T00407 CK9O6W 72705811 IC50 = 6309.57 nM T00407 CIW9K7 72713634 IC50 = 66000 nM T00407 C3W5VQ 72713635 IC50 = 74000 nM T00407 CBS16L 72713636 IC50 = 28000 nM T00407 C1LUB0 72713637 IC50 = 42000 nM T00407 C1Q6MO 72945553 IC50 = 290 nM T00407 C97BCW 72945554 IC50 = 74 nM T00407 CEW3O7 72945555 IC50 = 250 nM T00407 CL7EB1 73347805 IC50 = 91 nM T00407 CBD0N5 73349345 IC50 = 72 nM T00407 CUG1T8 73350913 IC50 = 29 nM T00407 CEH74A 73350914 IC50 = 42 nM T00407 C2C0ZX 73352391 IC50 = 398.11 nM T00407 C9VQ7H 73352402 IC50 = 1500 nM T00407 CD9NK1 73353867 IC50 = 380 nM T00407 CJY67C 73355395 IC50 = 2500 nM T00407 C3LQ4W 73425805 IC50 = 20 nM T00407 C2WDM8 73891130 IC50 = 1 nM T00407 C6VDW2 75373087 IC50 = 107410 nM T00407 CQOV07 75375570 IC50 > 200000 nM T00407 CW5A7G 76070631 IC50 = 126 nM T00407 CFZ65N 76071650 IC50 = 8 nM T00407 C0FD7H 76071652 IC50 = 15 nM T00407 CC3OJ7 76072013 IC50 = 9 nM T00407 CS7U4H 76072259 IC50 = 5 nM T00407 CQ78NK 76310219 IC50 = 158.49 nM T00407 CM4J8Q 76317442 IC50 = 251.19 nM T00407 CIN36T 76318560 IC50 = 7000000 nM T00407 CM7TH3 76328466 IC50 = 5011.87 nM T00407 C0T5NK 76335637 IC50 = 1000 nM T00407 CW7BS4 76534645 IC50 = 18 nM T00407 C9NE5G 76683426 IC50 = 30 nM T00407 CW6MD3 76683643 IC50 = 80 nM T00407 C3NIR2 76902013 IC50 = 37 nM T00407 CLW3A6 76902201 IC50 = 49 nM T00407 C46HRP 76902203 IC50 = 190 nM T00407 CKT41J 77108173 IC50 = 20 nM T00407 C8FRL6 77108189 IC50 = 10 nM T00407 CU6O0X 77461280 IC50 < 50 nM T00407 C5TB9S 77843982 Ki = 34 nM T00407 CI87ZD 77844001 IC50 = 1 nM T00407 CS6XE0 77846025 Ki = 12.2 nM T00407 COZ8S1 78319129 Ki = 77 nM T00407 C2TG5M 78320028 IC50 = 10 nM T00407 CTGH72 78320336 IC50 = 10 nM T00407 C85MTQ 78320816 Ki = 180 nM T00407 CCW9M4 78320817 Ki = 12 nM T00407 CN54HC 78321130 IC50 = 1.8 nM T00407 CX78QI 78321451 Ki = 43 nM T00407 CJA4F5 78322398 Ki = 47.8 nM T00407 CDZK41 78322399 Ki = 201 nM T00407 CZP9K2 78322539 IC50 = 140 nM T00407 CR6B4F 78323579 IC50 = 30 nM T00407 C3G2YK 78323818 IC50 = 20 nM T00407 C6BE7U 78325043 IC50 = 78 nM T00407 C4IF8T 78425807 Ki = 0.62 nM T00407 CVF12D 78428091 IC50 = 14 nM T00407 C4X6VZ 82104609 IC50 = 780 nM T00407 C4LA6F 86208116 IC50 = 637 nM T00407 CQUO30 86270617 Ki = 450 nM T00407 C1YFW8 86270651 Ki = 7.1 nM T00407 CHKW02 86270831 Ki = 26 nM T00407 CHK64J 86270834 Ki = 0.87 nM T00407 CFE7R3 86270928 Ki = 0.73 nM T00407 CE1V5Z 86270929 Ki = 16 nM T00407 C5KG4I 86271129 IC50 = 3.7 nM T00407 CT6BG3 86271751 Ki = 84 nM T00407 C81AKZ 86271752 EC50 = 280 nM T00407 C5WKC6 86271987 IC50 = 8 nM T00407 CV3YT8 86273096 IC50 = 27 nM T00407 CWPU56 86273098 IC50 = 31 nM T00407 C3EN0I 86273586 IC50 = 34 nM T00407 CB9AL4 86287631 IC50 < 11 nM T00407 CS4QR8 86287687 Ki = 120 nM T00407 C7SNT4 86287688 Ki = 17 nM T00407 CI8BA9 86287690 Ki = 11 nM T00407 COA7X4 86287755 Ki = 5.5 nM T00407 CB8JP3 86287958 Ki = 11 nM T00407 CDG13U 86295201 Ki = 54 nM T00407 C5M8RB 86295909 IC50 < 200 nM T00407 C8ONF2 86296101 IC50 = 35 nM T00407 CFV1S8 86296389 IC50 < 14 nM T00407 CX0KF8 86299084 Ki = 38 nM T00407 CS9F7V 86299086 Ki = 450 nM T00407 C9XR0G 86299218 Ki = 270 nM T00407 CUE87M 86299220 Ki = 1600 nM T00407 C6RT3M 86299506 EC50 > 10000 nM T00407 CXFG10 86301666 Ki = 3.8 nM T00407 C9W1SR 86581390 Ki = 1.3 nM T00407 CRN51L 86581538 Ki = 0.6 nM T00407 CE7B1X 86582295 IC50 = 3 nM T00407 C7IPH4 86582916 Ki = 2.1 nM T00407 C53QEW 86669224 IC50 = 6309.57 nM T00407 C7ZDO0 86808440 IC50 = 33160 nM T00407 C0RD6L 87056019 IC50 = 20 nM T00407 CQC6V8 87397080 IC50 > 100000 nM T00407 CY7P2N 89656146 Ki = 13 nM T00407 CW7PG2 89656147 IC50 = 58 nM T00407 C4JXL8 89656405 Ki = 680 nM T00407 CMSH53 89657387 Ki = 38 nM T00407 CGE9F1 89657420 Ki = 32 nM T00407 CEDL57 89657555 EC50 = 2480 nM T00407 CRU32W 89657560 Ki = 1.3 nM T00407 C8FXA7 89657583 Ki = 1.2 nM T00407 C1FOK3 90016835 Ki = 7 nM T00407 CXD3A6 90017103 EC50 = 370 nM T00407 CV8R0Z 90017113 Ki = 230 nM T00407 CUR5Z8 90017358 Ki = 22 nM T00407 CCB43O 90018193 Ki = 5.1 nM T00407 CZ54IL 90019075 Ki = 5.5 nM T00407 C2XQD4 90019266 Ki = 16 nM T00407 C4YE1K 90019789 Ki = 71 nM T00407 C8GN5H 90019850 Ki = 110 nM T00407 CV41WZ 90019957 Ki = 1900 nM T00407 CHK91R 90020090 Ki = 9 nM T00407 CU6CZ1 90026274 Ki = 450 nM T00407 CO82NI 90026512 Ki = 1700 nM T00407 CN4MG2 90026969 Ki = 890 nM T00407 CHC5I8 90027770 Ki = 13 nM T00407 C0T5SJ 90028262 Ki = 120 nM T00407 C13BOQ 90032394 Ki = 1700 nM T00407 CLQN32 90104652 IC50 = 10100 nM T00407 C68NDT 90364429 IC50 = 77 nM T00407 CPOG43 90387291 Ki = 41 nM T00407 CP25VC 90387467 Ki = 194 nM T00407 CZJ8W9 90387575 Ki = 16.1 nM T00407 C3JXP5 90387666 Ki = 98.1 nM T00407 C1EJ7F 90387844 IC50 = 200 nM T00407 CSW41E 90387917 Ki = 478 nM T00407 CW4IF5 90388035 Ki = 116 nM T00407 CED71H 90388046 Ki = 2182 nM T00407 C37YQH 90388075 Ki = 1948 nM T00407 C3C7GD 90388178 Ki = 1500 nM T00407 C6O2BH 90388309 Ki = 80 nM T00407 C1HD8T 90388367 Ki = 867 nM T00407 CFAE47 90388486 Ki = 98.8 nM T00407 C01MOG 90388523 Ki = 8322 nM T00407 CICK10 90388552 Ki = 824 nM T00407 CX90PZ 90395609 Ki = 19.7 nM T00407 C0UEK8 90395610 Ki = 18.5 nM T00407 CEYR46 90395611 Ki = 41.2 nM T00407 C5WG4S 90395612 Ki = 335 nM T00407 CHK85V 90395617 Ki < 0.5 nM T00407 CME05X 90395619 Ki < 0.5 nM T00407 C3WS5V 90395622 Ki = 30.6 nM T00407 C2D0LZ 90395625 Ki = 1.1 nM T00407 CNZ1V4 90395627 Ki = 7 nM T00407 CS4P9H 90395630 Ki = 44.3 nM T00407 CD94HJ 90395631 Ki = 2.8 nM T00407 CV75CK 90395632 IC50 > 1000 nM T00407 C62DJX 90395643 Ki = 22.5 nM T00407 C5XRI2 90395644 Ki = 4.2 nM T00407 CMX16I 90395646 Ki = 2.7 nM T00407 CQB83M 90395649 Ki = 2.8 nM T00407 CVK1M3 90395718 Ki = 52.3 nM T00407 CI28DM 90395720 Ki = 3.8 nM T00407 CW94AZ 90395721 Ki = 3.1 nM T00407 CYMD60 90395722 Ki = 42.6 nM T00407 C8UC4Z 90395724 Ki = 4.2 nM T00407 C1PJX2 90395725 Ki = 26.9 nM T00407 C49IVE 90395727 Ki = 139 nM T00407 C1KPZ5 90395734 Ki = 1.6 nM T00407 CFQ92A 90395738 Ki = 58.2 nM T00407 CR70LI 90395752 Ki = 1.4 nM T00407 C20LRN 90413429 Ki = 420 nM T00407 CLMV91 90413480 EC50 = 280 nM T00407 C3LC7M 90415492 Ki = 280 nM T00407 CD1Q4I 90417643 Ki = 17 nM T00407 CCF4T3 90466145 IC50 < 200 nM T00407 C1I7QN 90654869 IC50 > 30000 nM T00407 C1A6EO 90654871 IC50 = 7550 nM T00407 CCAL04 90654872 IC50 = 3180 nM T00407 C8F4IL 90667393 IC50 = 1995.26 nM T00407 CC76KI 90667394 IC50 = 1584.89 nM T00407 C07UWH 90667395 IC50 = 63095.73 nM T00407 CI79XN 90667396 IC50 = 19952.62 nM T00407 CYQ91J 90667397 IC50 = 6309.57 nM T00407 C4WCZ6 90667398 IC50 = 31622.78 nM T00407 C1J9HN 90667399 IC50 = 19952.62 nM T00407 C3WIR5 90667400 IC50 = 6309.57 nM T00407 CX1A3E 90667401 IC50 = 6309.57 nM T00407 C6FA3S 90667402 IC50 = 6309.57 nM T00407 CBS30L 90667403 IC50 = 3981.07 nM T00407 CV6DO1 90667404 IC50 = 630.96 nM T00407 C95ZKF 90667405 IC50 = 1258.93 nM T00407 CZP13T 90667406 IC50 = 794.33 nM T00407 CIA7N6 90667407 IC50 = 1000 nM T00407 CEA70Y 90667408 IC50 = 1584.89 nM T00407 C40KGW 90667409 IC50 = 794.33 nM T00407 CPMJ06 90667410 IC50 = 794.33 nM T00407 C64QIN 90667411 IC50 = 630.96 nM T00407 C83ORG 90667412 IC50 = 12589.25 nM T00407 C03DRI 90667413 IC50 = 1000 nM T00407 C16WGN 90667414 IC50 = 3981.07 nM T00407 CO92PS 90667415 IC50 = 10000 nM T00407 CLV2G0 90667416 IC50 = 1258.93 nM T00407 CJQZ54 90667417 IC50 = 630.96 nM T00407 CDRA20 90667418 IC50 = 1995.26 nM T00407 C0RX4B 90667452 IC50 = 50 nM T00407 C8HL5V 90667453 IC50 = 290 nM T00407 C3IE7F 90667454 IC50 = 360 nM T00407 C37GOB 90667455 IC50 = 100 nM T00407 C3PFG1 90670355 IC50 = 1690 nM T00407 C08KZL 90670356 IC50 = 15100 nM T00407 CD3P8Y 91215896 IC50 = 16000 nM T00407 CZ39RM 91668224 IC50 < 300 nM T00407 CYF7O2 91668539 IC50 = 50.12 nM T00407 C2JXG5 91668540 IC50 = 2511.89 nM T00407 CZ0H2Y 91668542 IC50 = 19952.62 nM T00407 C1BOU8 91758311 IC50 = 9 nM T00407 CB7Q8G 91809474 IC50 = 1400 nM T00407 CD7P5Y 91809475 IC50 = 250 nM T00407 CJ35EM 91809476 IC50 = 60 nM T00407 C8WX4I 91810827 IC50 < 5 nM T00407 CHOS65 91820723 IC50 = 25118.86 nM T00407 C0TNJ7 91820724 IC50 = 3981.07 nM T00407 C0N1GO 91826363 IC50 = 15 nM T00407 C8XL0I 91826394 IC50 < 11 nM T00407 CAZ9M0 91826677 IC50 = 3981.07 nM T00407 CEN52P 91826678 IC50 = 6309.57 nM T00407 CD0W7N 91971372 IC50 = 350 nM T00407 CY1WR2 92019884 IC50 = 2120000 nM T00407 C9WB3G 95828281 IC50 = 60000 nM T00407 CJ4MO9 95991007 IC50 > 100000 nM T00407 C3BIT0 100922929 IC50 = 90000 nM T00407 CU62EH 101481444 Ki = 25000 nM T00407 CB19IE 102358573 IC50 = 13000 nM T00407 CU91GC 105539824 IC50 = 26000 nM T00407 COD1I8 105539836 IC50 = 2580 nM T00407 C3M4CS 105539837 IC50 = 450 nM T00407 C3L5KU 105539840 IC50 = 450 nM T00407 C15PLR 105539841 IC50 = 2290 nM T00407 C9L7AG 105539842 IC50 = 730 nM T00407 CMDU18 105539860 IC50 = 410 nM T00407 C1W3XP 112499930 IC50 = 1900 nM T00407 CYX7T2 117072549 IC50 > 100000 nM T00407 C6EKA2 117689397 IC50 = 79 nM T00407 C4L1MR 117689434 IC50 = 107 nM T00407 CM9H5G 117689436 IC50 = 76 nM T00407 CUA1Z2 117689648 IC50 = 148 nM T00407 C8C6GE 117772437 Ki = 1.1 nM T00407 C5RF3K 117775483 Ki = 1.7 nM T00407 C24ZCQ 117775856 Ki = 0.6 nM T00407 C1RSV4 117833983 IC50 > 100000 nM T00407 C3PIB1 117833991 IC50 = 11800 nM T00407 CXL1W7 117834061 IC50 = 807 nM T00407 CG0LW1 117834596 IC50 = 968 nM T00407 C4OYH6 117834599 IC50 > 100000 nM T00407 C2QDF9 117834602 IC50 = 2890 nM T00407 CHF9V8 117834605 IC50 = 2760 nM T00407 C6B0TG 117834606 IC50 = 904 nM T00407 C0TLH3 117834615 IC50 = 474 nM T00407 CNJ58G 117834616 IC50 = 11000 nM T00407 CXK54D 117834619 IC50 = 3890 nM T00407 CN15HA 117834638 IC50 = 31500 nM T00407 CA0RF9 117834640 IC50 = 1660 nM T00407 C4K3JM 117834641 IC50 = 18800 nM T00407 CP8NJ4 117834648 IC50 = 4530 nM T00407 CE2TK1 117841251 IC50 = 13000 nM T00407 C0WZL6 117841252 IC50 = 12900 nM T00407 CH0L6O 117841253 IC50 = 51900 nM T00407 CD6H0A 117841254 IC50 = 13000 nM T00407 CVM0I2 117841255 IC50 = 562 nM T00407 C2JD5A 117841259 IC50 = 1170 nM T00407 CXVE97 117841261 IC50 = 479 nM T00407 C7PS8I 117841263 IC50 = 2050 nM T00407 CCU4G9 117841264 IC50 = 3170 nM T00407 CHS4W1 117841265 IC50 = 11900 nM T00407 CAK0P3 117841267 IC50 = 1620 nM T00407 C8YK5G 117841268 IC50 = 20700 nM T00407 CH6MJ5 117841269 IC50 = 2860 nM T00407 CP8KY3 117841270 IC50 = 860 nM T00407 C1NFO3 117891931 IC50 = 12 nM T00407 C4O8MX 117928476 IC50 < 1000 nM T00407 CV9T2S 118021357 IC50 = 420 nM T00407 C20BJO 118021398 IC50 = 920 nM T00407 CF1V6O 118021399 IC50 = 410 nM T00407 CA82SI 118021476 IC50 = 15 nM T00407 C9TJD6 118021554 IC50 = 9500 nM T00407 C7V1TN 118021622 IC50 = 2990 nM T00407 C3GM0W 118021678 IC50 = 24 nM T00407 C3BR8O 118021718 IC50 = 2 nM T00407 CDCF34 118021720 IC50 = 50 nM T00407 CSW7D8 118021721 IC50 = 510 nM T00407 C3LAW9 118021764 IC50 = 710 nM T00407 C4SCT5 118021773 IC50 = 460 nM T00407 C1IY8X 118021799 IC50 = 150 nM T00407 CD1P6E 118021813 IC50 = 2890 nM T00407 CGPK87 118021821 IC50 = 25 nM T00407 C72DWE 118021851 IC50 = 270 nM T00407 CA5CO3 118021879 IC50 = 160 nM T00407 CCR09V 118021930 IC50 = 368 nM T00407 CEG49X 118021977 IC50 = 750 nM T00407 C4JE7G 118021984 IC50 = 150 nM T00407 CF9YQ2 118022046 IC50 = 13000 nM T00407 CXAC70 118022070 IC50 = 240 nM T00407 C48NXS 118022125 IC50 = 49 nM T00407 C2MSO5 118022126 IC50 = 20000 nM T00407 C80GPR 118022184 IC50 = 250 nM T00407 C57CSH 118022209 IC50 = 240 nM T00407 C06EWP 118022266 IC50 = 1600 nM T00407 C7M9BE 118022285 IC50 = 11500 nM T00407 C97LFH 118022380 IC50 = 5 nM T00407 C8EGS1 118022691 IC50 = 3 nM T00407 C0MU6N 118022972 IC50 = 910 nM T00407 CUL98O 118060057 IC50 < 1000 nM T00407 CR15YL 118078883 IC50 = 370 nM T00407 CHDQ27 118078887 IC50 = 380 nM T00407 CN73AQ 118078912 IC50 = 43000 nM T00407 C6ZD3F 118078985 IC50 = 1600 nM T00407 CW6D8E 118079032 IC50 = 1400 nM T00407 C68LAH 118079235 IC50 = 60 nM T00407 CQJ6E2 118079293 IC50 < 100 nM T00407 C8S3BF 118079489 IC50 = 380 nM T00407 C9D8FA 118079501 IC50 = 100 nM T00407 CHP05V 118079652 IC50 = 420 nM T00407 CWN5B3 118079664 IC50 > 50000 nM T00407 C6VF5A 118079690 IC50 = 1600 nM T00407 CQ03GL 118079722 IC50 > 25000 nM T00407 CQ0BM1 118079985 IC50 > 50000 nM T00407 CIE48C 118080085 IC50 = 760 nM T00407 CU74JC 118080153 IC50 = 1700 nM T00407 CS1N3M 118080263 IC50 = 14000 nM T00407 C7D8OM 118080305 IC50 = 790 nM T00407 C6IJZ3 118080562 IC50 = 260 nM T00407 CMU0G5 118093990 IC50 = 1218 nM T00407 C61SNT 118094033 IC50 = 342 nM T00407 C0QT8P 118094069 IC50 = 596 nM T00407 C3G1DO 118116651 IC50 = 2.3 nM T00407 CLJ43Y 118117152 IC50 = 11 nM T00407 C6A1RW 118120978 IC50 = 10120 nM T00407 CHB87O 118120979 IC50 = 2890 nM T00407 CQ5V6F 118121011 IC50 = 4960 nM T00407 C5RS9G 118137754 Ki = 8.9 nM T00407 CZH8X7 118137759 Ki = 1.5 nM T00407 CYA1M0 118137762 IC50 = 2 nM T00407 CBGI40 118137765 Ki = 11 nM T00407 C29BNE 118137780 Ki = 1.9 nM T00407 CAB1X0 118137789 Ki = 1.5 nM T00407 CH9Z3Y 118137820 Ki = 2.8 nM T00407 C8A0CL 118137846 Ki = 3.4 nM T00407 CT8J9Y 118137861 Ki = 7.3 nM T00407 C8P3YF 118137879 Ki = 100 nM T00407 CGQY32 118137892 Ki = 3.8 nM T00407 CR0H9F 118137913 Ki = 2 nM T00407 CM06ZO 118138005 Ki = 0.8 nM T00407 C5Q4MC 118138006 IC50 = 1.3 nM T00407 C5P9RD 118169070 IC50 < 150 nM T00407 CAD1B6 118196369 IC50 < 5 nM T00407 CK50FQ 118196502 IC50 < 5 nM T00407 CPTF61 118200167 IC50 = 13900 nM T00407 CJ8YA2 118200170 IC50 = 5900 nM T00407 CZAI75 118200236 IC50 = 1940 nM T00407 C4Y5DB 118237331 IC50 = 63 nM T00407 C4P7MG 118277818 Ki = 27 nM T00407 CZ7D5J 118288035 IC50 = 150 nM T00407 CKG9S0 118288047 Ki = 99 nM T00407 C8ZQL1 118288049 Ki = 470 nM T00407 CGR63N 118288050 IC50 = 100 nM T00407 C73MQC 118317783 IC50 = 650 nM T00407 C5VQM0 118340530 Ki = 21.5 nM T00407 CG7WB4 118340538 Ki = 0.5 nM T00407 C13IJX 118340548 Ki = 2.6 nM T00407 C90KHI 118340551 Ki = 2 nM T00407 CS1D3I 118340553 Ki = 387 nM T00407 C6T9PS 118340596 Ki = 16.7 nM T00407 CQD5U2 118340603 Ki = 0.7 nM T00407 CR26LY 118340612 Ki < 1 nM T00407 CX09DZ 118340631 IC50 > 1000 nM T00407 C25VBU 118340646 Ki = 78 nM T00407 CI6E9H 118340650 Ki = 3.4 nM T00407 CZN8G5 118340653 Ki = 66.5 nM T00407 CFH02N 118340663 Ki < 1 nM T00407 C5T2HE 118340668 Ki = 2.4 nM T00407 CZT5M4 118340676 Ki = 6.3 nM T00407 C3RM5Q 118340684 Ki < 1 nM T00407 COR5G3 118340697 Ki = 1.7 nM T00407 C0GJZ5 118340710 Ki = 15.8 nM T00407 CF2C0W 118340714 Ki = 77.9 nM T00407 CM5TN1 118340720 Ki < 1 nM T00407 CXVK68 118340726 Ki = 3.1 nM T00407 CM34GO 118340729 Ki < 1 nM T00407 CPI9J0 118340741 Ki = 31 nM T00407 CS8KG3 118340760 Ki = 0.8 nM T00407 C35BHR 118340789 Ki = 28.4 nM T00407 C7IAX1 118340796 Ki = 1.2 nM T00407 C1MHG0 118340829 Ki = 1 nM T00407 CN1K0V 118340834 Ki = 4.9 nM T00407 C60DGX 118340843 Ki < 1 nM T00407 CE58WP 118509530 IC50 = 1.3 nM T00407 CXT73W 118509541 IC50 = 5 nM T00407 C8ZLN9 118693661 IC50 = 1.7 nM T00407 CR0PO8 118693673 Ki = 1.585 nM T00407 C8YNI5 118693928 Ki = 3.981 nM T00407 CPN74M 118719856 IC50 = 794.33 nM T00407 CE8DL3 118719857 IC50 = 630.96 nM T00407 COEU47 118719858 IC50 = 1000 nM T00407 CX05SW 118719859 IC50 = 630.96 nM T00407 CRCG07 118719860 IC50 = 501.19 nM T00407 C03XDG 118719861 IC50 = 501.19 nM T00407 C3ML2F 118719862 IC50 = 794.33 nM T00407 CZ67WF 118719863 IC50 = 25118.86 nM T00407 C0HR9Y 118719864 IC50 = 630.96 nM T00407 C7F4EP 118719865 IC50 = 316.23 nM T00407 CA40QV 118719866 IC50 = 630.96 nM T00407 CZ8QI6 118719867 IC50 = 794.33 nM T00407 C8NRI9 118719868 IC50 = 1000 nM T00407 C3Y2WT 118719869 IC50 = 1000 nM T00407 C52HPM 118719870 IC50 = 501.19 nM T00407 CUT97H 118719871 IC50 = 630.96 nM T00407 CBE68N 118719872 IC50 = 1000 nM T00407 C29WRE 118719873 IC50 = 794.33 nM T00407 C8J0TY 118719874 IC50 = 1000 nM T00407 CZR10C 118719875 IC50 = 3981.07 nM T00407 C35AWU 118719876 IC50 = 2511.89 nM T00407 C4OFG7 118721302 IC50 = 16300 nM T00407 CA8HW2 118721303 IC50 > 100000 nM T00407 CZY31K 118721304 IC50 > 50118.72 nM T00407 CYGS87 118721305 IC50 = 1584.89 nM T00407 C9O0IC 118721631 IC50 = 69900 nM T00407 CE9Y5W 118721632 IC50 = 7860 nM T00407 C63SEK 118727389 IC50 = 17900 nM T00407 C8NWB4 118727390 IC50 = 7800 nM T00407 C7F9XN 118727392 IC50 = 7200 nM T00407 C90BQI 118727394 IC50 = 78600 nM T00407 C9YJN5 118727397 IC50 = 63000 nM T00407 C8LA9O 118727400 IC50 = 29700 nM T00407 C6YUB8 118727401 IC50 = 20000 nM T00407 CGL92E 118727402 IC50 = 5600 nM T00407 CA82PM 118727403 IC50 = 427 nM T00407 CI4CQ2 118732060 IC50 = 2260 nM T00407 CIGL03 118732061 IC50 = 2060 nM T00407 C4ZA8M 118732062 IC50 > 10000 nM T00407 CQ71XK 118732063 IC50 = 8330 nM T00407 C8TRM7 118732064 IC50 = 7340 nM T00407 C6Z5CE 118732065 IC50 > 10000 nM T00407 CEXW89 118732066 IC50 > 10000 nM T00407 CTDN06 118732067 IC50 = 9310 nM T00407 CR07PK 118732068 IC50 = 5820 nM T00407 CJG89V 118732069 IC50 = 220 nM T00407 CDV60F 118732070 IC50 = 760 nM T00407 CFVW10 118732071 IC50 = 500 nM T00407 CAFB70 118732072 IC50 = 120 nM T00407 CN6D1A 118732073 IC50 = 400 nM T00407 CV3U7I 118732074 IC50 = 800 nM T00407 CM5YS0 118732075 IC50 = 300 nM T00407 CJWX45 118732076 IC50 = 60 nM T00407 CX35ZI 118732077 IC50 = 460 nM T00407 CQ84KV 118732078 IC50 = 140 nM T00407 CF57ZY 118732079 IC50 = 220 nM T00407 CL6U1T 118732080 IC50 = 170 nM T00407 C0XIA1 118732081 IC50 = 930 nM T00407 C7V9JG 118732082 IC50 = 100 nM T00407 CS2V9Y 118732083 IC50 = 790 nM T00407 CA3S1C 118732084 IC50 = 250 nM T00407 CU95AV 118740117 IC50 > 84000 nM T00407 C87ZPY 118796358 IC50 > 100000 nM T00407 CRF4G8 118796361 IC50 = 1121 nM T00407 CWS6Y5 118796362 IC50 = 3681 nM T00407 C9VQX4 118863284 IC50 = 0.7 nM T00407 C38TSJ 118863314 IC50 = 4.6 nM T00407 CQ2GC8 118863432 Ki = 7.3 nM T00407 CE4PK9 118863469 Ki = 4.1 nM T00407 CF9J8E 118918705 IC50 = 1700 nM T00407 CA3Z8O 118918714 IC50 = 2800 nM T00407 C8GLJ3 118918720 IC50 = 7200 nM T00407 C2ZY3U 118932975 IC50 > 10000 nM T00407 CC14FI 118933132 IC50 = 4500 nM T00407 CGO91Y 118933136 IC50 = 17000 nM T00407 CFMJ96 119081417 IC50 = 2900 nM T00407 C8AZ4C 119081691 IC50 = 2500 nM T00407 CUWX94 119081692 IC50 = 65 nM T00407 C9MQF0 119098887 IC50 = 30652 nM T00407 C0QX4D 119098889 IC50 = 23576 nM T00407 CBD7I6 121232405 IC50 = 19952.62 nM T00407 C4JN5Q 121237855 IC50 = 2400 nM T00407 C4AU0X 121237856 IC50 > 120000 nM T00407 C7A2UY 121237857 IC50 = 1500 nM T00407 CBN53Q 121271705 IC50 = 8500 nM T00407 CGBI67 121271742 IC50 = 13000 nM T00407 CPU76D 121271756 IC50 > 20000 nM T00407 CN4X9G 121271781 IC50 = 8900 nM T00407 CB83MK 121271792 IC50 = 11000 nM T00407 C0F6MH 121277645 IC50 > 200000 nM T00407 C0FA3C 121277864 IC50 = 16000 nM T00407 CP1NH2 121277975 IC50 = 4500 nM T00407 C0XVY8 121277987 IC50 = 8000 nM T00407 CHO97R 121277993 IC50 = 12000 nM T00407 COW87E 121278062 IC50 = 7000 nM T00407 C1PGY8 121278155 IC50 > 20000 nM T00407 C3GD2W 121335190 IC50 = 460 nM T00407 C81OYL 121335218 IC50 > 20000 nM T00407 C83RUE 121335260 IC50 = 8200 nM T00407 CECP26 121335281 IC50 = 1500 nM T00407 C1HR3M 121335283 IC50 > 20000 nM T00407 C2EP5S 121335312 IC50 = 2300 nM T00407 CNW25A 121338193 IC50 = 6100 nM T00407 C5JYP8 121338332 IC50 > 20000 nM T00407 C5ML2V 121338401 IC50 > 20000 nM T00407 C3JMB8 121338437 IC50 > 20000 nM T00407 CF25LT 121338490 IC50 > 20000 nM T00407 C5US9K 121338530 IC50 = 19200 nM T00407 CMF5D4 121338574 IC50 = 17200 nM T00407 C0VF7X 121338589 IC50 > 20000 nM T00407 CQ30XW 121342392 IC50 = 3600 nM T00407 CNM34X 121342393 IC50 = 3400 nM T00407 CXI0K8 121342398 IC50 = 600 nM T00407 C9O4RD 121342404 IC50 = 1200 nM T00407 CJMF61 121342523 IC50 = 1800 nM T00407 CQKU78 121342528 IC50 = 7900 nM T00407 C8CV7M 121365342 IC50 > 20000 nM T00407 C41LZU 121365398 IC50 = 18000 nM T00407 CNJ4A0 121365442 IC50 = 8500 nM T00407 C12KNG 121365488 IC50 = 3700 nM T00407 C8YE5F 121365519 IC50 = 3100 nM T00407 C46MHD 121372830 IC50 = 4200 nM T00407 CIW10X 121372875 IC50 = 7300 nM T00407 CFH51D 121372877 IC50 = 5600 nM T00407 C7W2KQ 121372879 IC50 = 13000 nM T00407 C7P2EW 121372880 IC50 > 20000 nM T00407 CDC61P 121372884 IC50 = 5900 nM T00407 C34YHN 121372887 IC50 = 13000 nM T00407 C6EID7 121372897 IC50 > 20000 nM T00407 C94PWO 121372898 IC50 = 4600 nM T00407 CL67ME 121372914 IC50 = 7300 nM T00407 CQ8ZL9 121372939 IC50 = 20000 nM T00407 C3I8SV 121372947 IC50 = 9600 nM T00407 CKYL73 121372990 IC50 = 4200 nM T00407 CQ0AL8 121372997 IC50 = 4000 nM T00407 C32SNH 121373004 IC50 = 870 nM T00407 C4UD7J 121373027 IC50 = 6400 nM T00407 CV9KF4 121373031 IC50 > 20000 nM T00407 CE2VJ4 121373032 IC50 = 9200 nM T00407 CZ30EX 121373033 IC50 = 12000 nM T00407 C1HRP7 121373036 IC50 > 20000 nM T00407 CP0OX4 121373042 IC50 = 15000 nM T00407 CDQV23 121373043 IC50 = 13000 nM T00407 CVO7B2 121373072 IC50 = 2200 nM T00407 CD9PJ2 121373074 IC50 = 3900 nM T00407 C57ZDO 121373154 IC50 = 4600 nM T00407 CS9XW0 121373155 IC50 = 8600 nM T00407 CYDN26 121373156 IC50 = 3700 nM T00407 CI84KM 121373164 IC50 = 3800 nM T00407 CK03TO 121373206 IC50 = 16000 nM T00407 C4G2QK 121373220 IC50 > 20000 nM T00407 C57GXL 121373316 IC50 = 4100 nM T00407 C04UKS 121373365 IC50 = 5400 nM T00407 CDH8M4 121373418 IC50 = 4200 nM T00407 C1TK3U 121373476 IC50 > 20000 nM T00407 CW1HV7 121373599 IC50 = 11000 nM T00407 C2V6AX 121373769 IC50 = 9500 nM T00407 C47QXT 121376807 IC50 = 13000 nM T00407 C9XWC0 121376818 IC50 = 12000 nM T00407 C0QKG5 121376850 IC50 = 4800 nM T00407 CP6R5B 121382912 IC50 = 4000 nM T00407 C51UXY 121414852 IC50 = 160 nM T00407 C19VLJ 121414853 IC50 = 130 nM T00407 CL5SB9 121414854 IC50 = 15 nM T00407 CWC98G 121499171 IC50 = 25118.86 nM T00407 C6E0UL 122164589 Ki = 12.59 nM T00407 C5PKZ6 122164734 IC50 = 70 nM T00407 C67WYM 122164963 Ki = 7.943 nM T00407 CEF87B 122164964 Ki > 1000 nM T00407 CO9J5W 122179607 IC50 = 1258.93 nM T00407 C3WOE8 122179608 IC50 = 6309.57 nM T00407 CW03JY 122179609 IC50 = 1000 nM T00407 CHNS18 122179610 IC50 = 3162.28 nM T00407 C2Q0OY 122179611 IC50 = 1258.93 nM T00407 C9GPL4 122179612 IC50 = 6309.57 nM T00407 CZX41C 122179613 IC50 = 3981.07 nM T00407 CJDK15 122179614 IC50 = 7943.28 nM T00407 CSF76G 122179615 IC50 = 1995.26 nM T00407 CY7U0Z 122179616 IC50 = 794.33 nM T00407 C1MV9L 122179617 IC50 = 1258.93 nM T00407 CJ81BV 122179618 IC50 = 15848.93 nM T00407 CZ69QO 122180530 IC50 > 50118.72 nM T00407 C7D5VP 122180531 IC50 = 39810.72 nM T00407 CRY84E 122180532 IC50 = 5011.87 nM T00407 C0J1AY 122180533 IC50 = 50118.72 nM T00407 CPIV02 122180534 IC50 > 50118.72 nM T00407 CC9XH7 122180535 IC50 > 50118.72 nM T00407 C0IWE1 122180536 IC50 > 501187.23 nM T00407 CEF19P 122180537 IC50 = 10000 nM T00407 C20LOD 122180538 IC50 = 19952.62 nM T00407 C73OMU 122180539 IC50 = 6309.57 nM T00407 CZSB51 122180540 IC50 = 6309.57 nM T00407 CJ4LO2 122180541 IC50 = 15848.93 nM T00407 C4TB0F 122180542 IC50 = 10000 nM T00407 CTXL15 122180543 IC50 = 39810.72 nM T00407 CUDY80 122180544 IC50 = 12589.25 nM T00407 C0SC2Y 122180545 IC50 = 25118.86 nM T00407 CR6T4G 122180546 IC50 = 25118.86 nM T00407 CHJG86 122180547 IC50 = 158489.32 nM T00407 CYZV97 122180548 IC50 = 15848.93 nM T00407 C0AIU8 122180549 IC50 = 12589.25 nM T00407 CPUS31 122180550 IC50 = 12589.25 nM T00407 CD62RB 122180551 IC50 = 6309.57 nM T00407 C8UCV9 122180552 IC50 = 3162.28 nM T00407 C72NLB 122180553 IC50 = 5011.87 nM T00407 CR0K5P 122180554 IC50 = 7943.28 nM T00407 CZ6L2N 122180555 IC50 = 3981.07 nM T00407 CKH49I 122180556 IC50 = 3162.28 nM T00407 CS4PD6 122180557 IC50 = 794.33 nM T00407 CWC9I4 122180558 IC50 = 1000 nM T00407 CE7SL5 122180559 IC50 = 630.96 nM T00407 CR6YD4 122180560 IC50 = 125.89 nM T00407 C8HCK6 122180561 IC50 = 1995.26 nM T00407 CX9C6Y 122180562 IC50 = 794.33 nM T00407 CPZ67Y 122180563 IC50 = 3162.28 nM T00407 CN1LE0 122180564 IC50 = 5011.87 nM T00407 C4ITM8 122180892 IC50 = 13000 nM T00407 CFCA87 122180893 IC50 = 13000 nM T00407 CZRJ29 122180894 IC50 = 13000 nM T00407 C8RE2M 122180895 IC50 = 14000 nM T00407 C54NBV 122180896 IC50 = 16000 nM T00407 C26RAL 122180897 IC50 = 18000 nM T00407 CC35RW 122180898 IC50 = 25000 nM T00407 C7E3VM 122180899 IC50 = 25000 nM T00407 C2UQW0 122180900 IC50 = 34000 nM T00407 C67LPS 122180901 IC50 = 40000 nM T00407 C3FC0Z 122180902 IC50 = 44000 nM T00407 CSR48T 122180903 IC50 = 46000 nM T00407 CVI96R 122180904 IC50 > 50000 nM T00407 CZB15E 122180905 IC50 = 9000 nM T00407 C6V0UQ 122180906 IC50 = 13000 nM T00407 COR80H 122180907 IC50 = 25000 nM T00407 CFVN54 122180908 IC50 = 29000 nM T00407 CXP8T3 122180909 IC50 = 44000 nM T00407 CE29NL 122180910 IC50 = 47000 nM T00407 CR78FH 122180911 IC50 = 49000 nM T00407 CB1M0U 122180912 IC50 > 50000 nM T00407 CGLF82 122181547 IC50 = 6309.57 nM T00407 CZGK74 122181548 IC50 = 10000 nM T00407 C9P3GX 122181549 IC50 = 10000 nM T00407 C3QJ5L 122181550 IC50 = 15848.93 nM T00407 C3NC4V 122181552 IC50 = 7943.28 nM T00407 C41ZXJ 122181555 IC50 = 1584.89 nM T00407 C6I3VJ 122181557 IC50 = 630.96 nM T00407 C7CJR2 122181559 IC50 = 12589.25 nM T00407 CP5Z1C 122181560 IC50 = 15848.93 nM T00407 C61RTG 122181561 IC50 = 12589.25 nM T00407 CT62FG 122181571 IC50 = 10000 nM T00407 CJ8B1U 122187515 Ki = 7950 nM T00407 CHI14C 122187516 Ki = 4500 nM T00407 CUX72G 122187517 Ki > 10000 nM T00407 CI86PH 122187518 Ki > 10000 nM T00407 CD24VL 122187519 Ki = 1400 nM T00407 C8ZLB5 122187520 Ki > 10000 nM T00407 C6OGU0 122187521 Ki = 970 nM T00407 CW84YE 122187522 Ki = 8.7 nM T00407 CH83IY 122187523 Ki = 37 nM T00407 C6CWM2 122187524 Ki = 46 nM T00407 C24AKR 122187525 Ki = 29 nM T00407 CZ3E7H 122187526 Ki = 100 nM T00407 CO25IW 122191031 IC50 >= 10000 nM T00407 C4WGV6 122191040 IC50 = 4000 nM T00407 CDY43J 122191048 IC50 >= 10000 nM T00407 C79NTO 122446081 IC50 = 14 nM T00407 C0LNZ9 122446098 IC50 = 21 nM T00407 C5EQJ0 122467457 IC50 = 4290 nM T00407 C4ME9H 122467464 IC50 > 30000 nM T00407 C56NAS 122467465 IC50 = 4170 nM T00407 C35LXF 122467467 IC50 > 30000 nM T00407 CEJ5W3 122467468 IC50 = 3440 nM T00407 C80AFH 122467469 IC50 = 2550 nM T00407 C5BY0I 122467470 IC50 = 600 nM T00407 CO8R3Y 122467472 IC50 = 5640 nM T00407 C3E6UB 122467476 IC50 = 4840 nM T00407 CQ71FH 122467477 IC50 > 30000 nM T00407 C6V7LS 122467478 IC50 = 1210 nM T00407 C7QV4I 122467480 IC50 > 30000 nM T00407 C12RVQ 122467483 IC50 > 30000 nM T00407 CLAE37 122467484 IC50 = 1500 nM T00407 CY2CD5 122467486 IC50 = 510 nM T00407 CM4NH1 122467488 IC50 = 5290 nM T00407 COCT-54 122467494 IC50 > 30000 nM T00407 CKC3B1 122467495 IC50 = 4100 nM T00407 CNI3H2 122467498 IC50 = 1120 nM T00407 C62IDL 122470439 IC50 = 10 nM T00407 C7VJH3 122512239 IC50 = 12.59 nM T00407 C6DS2X 122553424 IC50 < 11 nM T00407 CU8L1O 122553479 IC50 = 12 nM T00407 CN51WG 122588588 IC50 < 0.5 nM T00407 C3C8QO 122588611 IC50 = 3 nM T00407 C0KE5N 122588642 IC50 = 2 nM T00407 CWJD15 122705990 IC50 > 10000 nM T00407 CIR48B 123146482 IC50 = 501.19 nM T00407 CR9T6N 123814574 IC50 = 1000 nM T00407 C7GWV1 124098192 IC50 = 18800 nM T00407 C5VQN1 124429951 IC50 = 3980 nM T00407 C20LTP 125383342 IC50 = 77 nM T00407 CR98TS 125994265 IC50 > 10000 nM T00407 C4GYP3 126521168 IC50 = 32 nM T00407 CL2PG5 126521180 IC50 = 18 nM T00407 CQV90I 126521354 IC50 = 28 nM T00407 C0HJV7 126521430 IC50 > 999 nM T00407 CN6FI1 126521537 IC50 = 2 nM T00407 C1DOG4 126521586 IC50 = 14 nM T00407 CRY0S6 126563516 IC50 = 12 nM T00407 CN0D6M 126563562 IC50 = 10 nM T00407 CKB36S 126563576 IC50 = 7 nM T00407 CX79NH 126563597 IC50 = 14 nM T00407 C2K5XG 126563611 IC50 = 17 nM T00407 CZ06NR 126563612 IC50 = 36 nM T00407 CM5P2Z 126563615 IC50 = 30 nM T00407 C15ILF 126564427 IC50 = 7 nM T00407 CROY39 126564463 IC50 = 7 nM T00407 CHO12Y 126564469 IC50 > 10000 nM T00407 CB2AS4 126564470 IC50 = 6 nM T00407 CBW08I 126564471 IC50 = 12 nM T00407 CD78GB 126564481 IC50 = 10 nM T00407 CU8CA9 126564486 IC50 = 6 nM T00407 CQW6P1 126564822 IC50 = 11 nM T00407 CQS5T2 126564831 IC50 = 23 nM T00407 CNP2L7 126564832 IC50 = 13 nM T00407 C58PNK 126564833 IC50 = 15 nM T00407 CHPV09 126564847 IC50 = 10 nM T00407 CJZW04 126564858 IC50 = 13 nM T00407 C4WXN8 126772498 IC50 = 24910 nM T00407 CM8EB4 126961333 IC50 = 16700 nM T00407 C0MR6T 126961716 Ki = 970 nM T00407 CJR0V7 127025419 IC50 = 1258.93 nM T00407 CZ93IW 127025420 IC50 = 398.11 nM T00407 C5FV9L 127025697 IC50 = 501.19 nM T00407 C8N5UA 127025979 IC50 = 2511.89 nM T00407 C7M2GL 127025980 IC50 = 15848.93 nM T00407 C2LYR4 127025981 IC50 = 12589.25 nM T00407 C8GLF2 127025982 IC50 = 199.53 nM T00407 CMG7C1 127026579 IC50 = 38900 nM T00407 C57IHP 127026582 IC50 > 50000 nM T00407 CF9QV5 127026591 IC50 > 50000 nM T00407 C4MY5E 127026593 IC50 > 50118.72 nM T00407 C7OQT2 127026594 IC50 = 1584.89 nM T00407 C62OFC 127026595 IC50 = 794.33 nM T00407 C0C1HZ 127028091 IC50 > 50000 nM T00407 COXV68 127029808 IC50 = 5560 nM T00407 CS37AQ 127030405 IC50 < 300 nM T00407 C0DF1I 127030450 IC50 > 30000 nM T00407 CV81XG 127030451 IC50 = 2980 nM T00407 CNG8Y1 127030726 IC50 = 85 nM T00407 C6B4HD 127030768 IC50 = 1580 nM T00407 C5XN8O 127030774 IC50 = 3510 nM T00407 C6FI7V 127031094 IC50 = 470 nM T00407 CB7X6C 127031095 IC50 = 3870 nM T00407 C7GQI0 127031954 IC50 = 1160 nM T00407 CEVK16 127032241 IC50 = 1670 nM T00407 CVOS94 127032857 IC50 = 3130 nM T00407 CH14FC 127032939 IC50 = 8100 nM T00407 CR2A7U 127033172 IC50 = 1190 nM T00407 C1SA9P 127033473 IC50 > 30000 nM T00407 C0P5EA 127033474 IC50 = 4270 nM T00407 CBT9C7 127033475 IC50 = 1170 nM T00407 C30AKN 127033476 IC50 = 460 nM T00407 CIG3Q9 127033567 IC50 = 20400 nM T00407 CS4NG8 127033568 IC50 = 26400 nM T00407 C0JYH2 127033770 IC50 = 210 nM T00407 CG20LF 127034058 IC50 = 4900 nM T00407 CCK36M 127034059 IC50 = 4810 nM T00407 C2JOB7 127034595 IC50 = 400 nM T00407 C3R6VW 127034596 IC50 = 620 nM T00407 CRH92V 127034597 IC50 = 1720 nM T00407 C7V0HE 127034598 IC50 = 120 nM T00407 CV07YO 127038801 IC50 <= 1000 nM T00407 C4RGQ7 127043287 IC50 > 50118.72 nM T00407 CF3Z9G 127043292 IC50 > 50118.72 nM T00407 CA3VI9 127043861 IC50 = 10000 nM T00407 CCSJ69 127043862 IC50 > 50118.72 nM T00407 CJT6N0 127043863 IC50 = 25118.86 nM T00407 CEG46M 127043864 IC50 = 7943.28 nM T00407 CL8S6X 127043872 IC50 > 50118.72 nM T00407 CEAN18 127043873 IC50 > 50118.72 nM T00407 CZP0D9 127043874 IC50 = 10000 nM T00407 C7Y1IB 127043875 IC50 = 12589.25 nM T00407 CH4BE8 127043876 IC50 > 50118.72 nM T00407 CWP65X 127043881 IC50 = 19952.62 nM T00407 CO62HW 127044040 IC50 = 39810.72 nM T00407 CE0CG1 127044041 IC50 > 50118.72 nM T00407 CJ7YT3 127044046 IC50 > 50118.72 nM T00407 CAN9K0 127044332 IC50 > 50118.72 nM T00407 CH1MJ8 127044333 IC50 > 50118.72 nM T00407 CP15DV 127044334 IC50 > 50118.72 nM T00407 CU7X9E 127044335 IC50 > 50118.72 nM T00407 CXN63Y 127044336 IC50 > 50118.72 nM T00407 CLN5S3 127044787 IC50 > 50118.72 nM T00407 CX4M3R 127044824 IC50 > 50118.72 nM T00407 CZ5H7K 127045294 IC50 = 10000 nM T00407 CQOL84 127045572 IC50 = 39810.72 nM T00407 CGA71L 127048256 IC50 = 61917 nM T00407 CH6T5J 127048257 IC50 = 67479 nM T00407 C60SZQ 127048258 IC50 = 47095 nM T00407 C6BT3U 127048317 IC50 > 20000 nM T00407 C9DY4Z 127048318 IC50 = 8000 nM T00407 C5AV7U 127049278 IC50 = 31421 nM T00407 C50BMV 127049279 IC50 = 5861 nM T00407 CTFY41 127049280 IC50 = 32430 nM T00407 CVE71A 127049281 IC50 = 19165 nM T00407 C73TND 127049282 IC50 = 3778 nM T00407 CEN16G 127049286 IC50 = 44000 nM T00407 C9C0MB 127049631 IC50 = 3500 nM T00407 C8MXQ7 127049932 IC50 > 20000 nM T00407 C2VC3L 127050405 IC50 = 1147 nM T00407 CWFM08 127050492 IC50 = 81300 nM T00407 CTF4N2 127051087 IC50 > 100000 nM T00407 CD2T1E 127051228 IC50 = 780 nM T00407 CPS8R6 127051229 IC50 = 850 nM T00407 C12KXI 127051477 IC50 > 20000 nM T00407 CRZ3A6 127051526 IC50 = 670 nM T00407 CR0P6Q 127051527 IC50 = 3730 nM T00407 CLSZ47 127051725 IC50 = 23005 nM T00407 CMY93U 127051726 IC50 = 47359 nM T00407 CY8V1A 127051727 IC50 > 100000 nM T00407 CXZT48 127052023 IC50 > 100000 nM T00407 C9V3AX 127052165 IC50 = 1490 nM T00407 C2OHP4 127052166 IC50 = 1380 nM T00407 CS60GZ 127052167 IC50 = 1050 nM T00407 C2RB3T 127052469 IC50 = 2990 nM T00407 CHA05V 127052470 IC50 = 770 nM T00407 C5EYK2 127053005 IC50 > 20000 nM T00407 CG6AY7 127053006 IC50 > 20000 nM T00407 CGM6W4 128963618 IC50 > 20000 nM T00407 CT2M0R 129214093 Ki = 10.4 nM T00407 C7C0WK 129606900 IC50 = 79.43 nM T00407 CO8Z2N 129900111 IC50 = 34000 nM T00407 CTLO82 130345485 Ki = 70 nM T00407 CJ6VO1 130345500 Ki = 190 nM T00407 C4DJO5 130345531 Ki = 1500 nM T00407 CIJ23L 130345532 Ki = 13 nM T00407 CX32JZ 130345556 Ki = 3300 nM T00407 CO0L1R 130345558 Ki = 15 nM T00407 C9L1OG 130345579 Ki = 2.3 nM T00407 COI68Y 130345587 Ki = 2800 nM T00407 C8JV7L 130345597 Ki = 820 nM T00407 C0RTS8 130345606 Ki = 4.2 nM T00407 C98WYE 130345614 Ki = 33 nM T00407 C1XDL5 130345617 Ki = 2.1 nM T00407 C5FUX9 130357671 Ki = 250 nM T00407 CG2RM3 130357741 Ki = 2.7 nM T00407 C7NEB1 130471695 IC50 > 10800 nM T00407 CLA09E 130471696 IC50 > 20000 nM T00407 CWNY27 130471723 IC50 > 12100 nM T00407 CXW1B4 130471724 IC50 > 14500 nM T00407 C1EN7A 130471730 IC50 > 13900 nM T00407 C2HD6P 130471733 IC50 = 14500 nM T00407 C5DFI7 130471761 IC50 > 20000 nM T00407 CDLE96 130471765 IC50 > 20000 nM T00407 C1C8OB 130471770 IC50 > 9500 nM T00407 CDC32I 130471775 IC50 > 14250 nM T00407 C3D7HE 130471777 IC50 > 20000 nM T00407 CFI30C 130471784 IC50 > 11450 nM T00407 C7TJA6 130471785 IC50 > 15000 nM T00407 CDUX50 130471789 IC50 > 15000 nM T00407 C8VAM6 130471790 IC50 > 12950 nM T00407 CN80UV 130471849 IC50 > 20000 nM T00407 CEV5I3 130471855 IC50 > 15000 nM T00407 CE1K3M 130471876 IC50 > 11900 nM T00407 CFTG42 130472058 IC50 > 9950 nM T00407 C5P2ED 130472268 IC50 > 15000 nM T00407 C7B6CZ 130472269 IC50 = 15500 nM T00407 CED70X 130472274 IC50 > 10000 nM T00407 CNUG19 131740828 Ki = 1100 nM T00407 CK0B6N 131985884 IC50 = 1700 nM T00407 CUN18W 132005225 IC50 = 10800 nM T00407 CD84OI 132005228 IC50 = 6000 nM T00407 C7ASP9 132005246 IC50 = 18800 nM T00407 CE89ZR 132010072 Ki = 1.3 nM T00407 C0W9DE 132010081 Ki = 6.9 nM T00407 C39MLW 132010085 Ki = 1.2 nM T00407 CKB6N5 132010104 Ki = 1.1 nM T00407 CYE3D7 132010164 Ki = 1 nM T00407 C7WP0Z 132010280 Ki = 1.1 nM T00407 CFN06J 132010408 Ki = 2 nM T00407 CH1Y7G 132010677 Ki = 0.6 nM T00407 CJ2I1C 132010719 Ki = 0.5 nM T00407 C8IAW3 132010913 Ki = 1.5 nM T00407 CHO97Q 132010929 Ki = 1.3 nM T00407 CE61QG 132154358 IC50 = 0.43 nM T00407 COE15M 132166121 IC50 = 5100 nM T00407 CGNQ49 132168874 IC50 = 19000 nM T00407 CHC6A0 132168907 IC50 = 12000 nM T00407 CRV1I6 132168917 IC50 = 3800 nM T00407 CB4X0G 132169005 IC50 = 8900 nM T00407 CX9U1Y 132169030 IC50 > 20000 nM T00407 CO7QW0 132169133 IC50 = 7800 nM T00407 CD8SE7 132169397 IC50 > 20000 nM T00407 CG4X6Z 132169416 IC50 = 14000 nM T00407 CV8F3O 132169466 IC50 > 20000 nM T00407 C7EHB4 132169581 IC50 = 7400 nM T00407 CI3HC8 132169624 IC50 = 12000 nM T00407 CF7H3C 132169928 IC50 = 6900 nM T00407 C7KUC2 132176755 IC50 > 20000 nM T00407 C6HQ0I 132181409 IC50 > 20000 nM T00407 C2S4IT 132181414 IC50 = 1100 nM T00407 C3MV7Y 132181499 IC50 = 3900 nM T00407 CM2K6Z 132181651 IC50 = 18000 nM T00407 CZW36J 132181706 IC50 > 20000 nM T00407 CVZ87Y 132181707 IC50 = 4100 nM T00407 CXVW94 132181717 IC50 > 20000 nM T00407 CG13LT 132186451 IC50 = 15000 nM T00407 CGC84J 132186467 IC50 > 20000 nM T00407 CB23YA 132186468 IC50 = 8500 nM T00407 C06KYU 132186469 IC50 = 3200 nM T00407 CI56DE 132186470 IC50 > 20000 nM T00407 COK17B 132186514 IC50 = 14000 nM T00407 CE3H2T 132186523 IC50 = 2500 nM T00407 CG5SN9 132186583 IC50 = 4700 nM T00407 CN90OX 132186586 IC50 = 14000 nM T00407 CAR2X5 132186700 IC50 = 2800 nM T00407 C5A3QS 132186701 IC50 = 3300 nM T00407 CKY07I 132186706 IC50 > 20000 nM T00407 C4DOU1 132186760 IC50 > 20000 nM T00407 CFB2X6 132186767 IC50 = 13000 nM T00407 CM6K0J 132186772 IC50 = 7700 nM T00407 CL29US 132186773 IC50 = 11000 nM T00407 CUH7W8 132186890 IC50 = 6700 nM T00407 CGDN94 132275066 IC50 = 12000 nM T00407 C5LQ2Y 132289425 IC50 = 2511.89 nM T00407 CL1FY9 132451787 IC50 = 5600 nM T00407 C9UGN7 132503236 IC50 = 2700 nM T00407 CN3P0M 132961531 IC50 = 76 nM T00407 CU0E6V 132992936 IC50 = 234.42 nM T00407 C51OUR 133053976 IC50 = 52 nM T00407 C16VTU 134132238 IC50 > 20000 nM T00407 C6V4WU 134132252 IC50 = 9800 nM T00407 C5SV3A 134132771 IC50 > 20000 nM T00407 CANC79 134133805 IC50 > 20000 nM T00407 CAI3J0 134134171 IC50 = 18000 nM T00407 CFZ94S 134135176 IC50 = 7700 nM T00407 CV7K2Z 134135271 IC50 > 20000 nM T00407 C9OC2T 134135428 IC50 = 7420 nM T00407 C26RIB 134135696 IC50 = 4600 nM T00407 C8SCT7 134137178 IC50 > 20000 nM T00407 C7RFZ1 134139020 IC50 = 5800 nM T00407 C72VXC 134140106 IC50 = 6250 nM T00407 COC34Y 134140792 IC50 = 8240 nM T00407 CE16SF 134142067 IC50 > 20000 nM T00407 CU1Y5M 134142603 IC50 = 2740 nM T00407 C8D3NS 134143236 IC50 = 11000 nM T00407 CY83MP 134143286 IC50 > 20000 nM T00407 C1NKU6 134144625 IC50 = 11230 nM T00407 C1KAR7 134146622 IC50 > 20000 nM T00407 CWZ0V3 134147360 IC50 > 20000 nM T00407 CC87ZT 134149739 IC50 > 20000 nM T00407 CA2HB7 134149861 IC50 > 20000 nM T00407 CF98TY 134149949 IC50 > 20000 nM T00407 CC29GZ 134151635 IC50 > 20000 nM T00407 CP51GS 134151910 IC50 > 20000 nM T00407 CIP61L 134153498 IC50 = 37000 nM T00407 C31JZR 134154313 IC50 > 20000 nM T00407 COX6Y9 134157699 IC50 = 14000 nM T00407 CBW6T0 134163707 IC50 = 283 nM T00407 CO3A0E 134817551 IC50 = 5011.87 nM T00407 CP4X5W 134817552 IC50 = 5011.87 nM T00407 CS7WX6 134821995 IC50 = 1000 nM T00407 CI2AM1 134828588 IC50 = 100 nM T00407 CJ9E8M 135121918 IC50 = 70 nM T00407 CS71IF 135126189 IC50 = 280 nM T00407 CK1BA5 135126537 IC50 = 2600 nM T00407 CRS95D 135126542 IC50 = 970 nM T00407 CZQ49P 135126546 IC50 = 520 nM T00407 CTO4K5 135143907 IC50 = 3900 nM T00407 CIAG86 135394452 IC50 > 20000 nM T00407 CRNY32 135397673 Ki = 0.5 nM T00407 C9J4PW 135398123 IC50 = 1990 nM T00407 C7L5ER 135398124 IC50 = 690 nM T00407 C9IGU4 135398125 IC50 = 630 nM T00407 CCTO31 135404086 IC50 = 4300 nM T00407 C39LZE 135404087 IC50 = 5200 nM T00407 CA40QW 135535536 IC50 > 50118.72 nM T00407 CV4X7R 135566898 Ki = 910 nM T00407 CU2F1G 135566900 Ki = 150 nM T00407 C5F3LV 135567026 IC50 = 430 nM T00407 CF8TQ2 135567084 IC50 = 1160 nM T00407 CZ84OQ 135567317 Ki = 10 nM T00407 CV2YA3 135630716 IC50 = 16000 nM T00407 CZK84G 135630721 IC50 = 31000 nM T00407 CKD1O7 135804260 IC50 = 4700 nM T00407 C4DMZ9 136002815 Ki = 6430 nM T00407 C6HJ9W 136174597 Ki = 6480 nM T00407 C0AY8G 136174600 Ki = 6830 nM T00407 CX9IM7 136174601 Ki = 520 nM T00407 CB26GV 136174603 Ki = 1300 nM T00407 CY4G3S 136174604 Ki = 1270 nM T00407 CQ02PC 136174605 Ki = 4670 nM T00407 CFH95M 136174610 Ki = 500 nM T00407 C4BO0T 136174611 Ki = 2790 nM T00407 CG9N5D 136174612 Ki = 1400 nM T00407 C69HZF 136174618 Ki = 7140 nM T00407 CWSG57 136212224 IC50 = 4310 nM T00407 C41NGO 136224170 Ki = 1280 nM T00407 CL7FQ1 136224171 Ki = 2310 nM T00407 C7O5PH 136226498 Ki = 4920 nM T00407 C1RH2I 136226499 Ki = 5970 nM T00407 CHY5I0 136226500 Ki > 100000 nM T00407 CYVZ61 136226501 Ki = 7120 nM T00407 CXJG97 136226502 Ki = 6130 nM T00407 CBHW80 136226503 Ki = 900 nM T00407 CWD47H 136226504 Ki = 320 nM T00407 CKPS21 136226505 Ki = 730 nM T00407 CP29FE 136226506 Ki = 6540 nM T00407 C81XIB 136226507 Ki = 9600 nM T00407 C9OJ6K 136226508 Ki = 1300 nM T00407 C6JRN2 136226509 Ki = 1840 nM T00407 CNT61S 136226510 Ki = 3130 nM T00407 CW94QO 136226511 Ki = 169.82 nM T00407 CAFU62 136226512 Ki = 6020 nM T00407 CFT26V 136226513 Ki = 2390 nM T00407 CJG3I4 136226514 Ki = 3910 nM T00407 C2PB9D 136242352 IC50 = 560 nM T00407 C27WOL 136244604 IC50 = 77000 nM T00407 CW8XN5 136321792 IC50 = 9280 nM T00407 CXLE13 136387525 Ki = 30 nM T00407 CFRV40 136387526 Ki = 37 nM T00407 CSPK74 136387543 Ki = 16 nM T00407 C4N2FR 136387545 Ki = 77 nM T00407 CY3UK2 136387556 Ki = 1100 nM T00407 CL6R5U 136387567 Ki = 150 nM T00407 C53FKI 136577469 IC50 = 6380 nM T00407 C0IY2P 136963109 IC50 < 100 nM T00407 C60DNA 137250528 IC50 = 11000 nM T00407 C6G9UA 137275811 IC50 = 328 nM T00407 CO71RI 137285009 IC50 = 32 nM T00407 CS9MR6 137285011 IC50 = 32 nM T00407 CL02HM 137319656 IC50 = 2092 nM T00407 C5E8GX 137319657 IC50 = 1416 nM T00407 CI1WA0 137319664 IC50 = 6600 nM T00407 C6ZG7K 137321201 IC50 = 501.19 nM T00407 CFXE14 137321203 IC50 = 50.12 nM T00407 CXN4U1 137321204 IC50 = 63.1 nM T00407 C6MGN1 137322665 IC50 = 32230 nM T00407 C31BFH 137347775 IC50 = 540 nM T00407 C7FVC0 137347776 IC50 = 260 nM T00407 CG8VK6 137348598 IC50 = 2000 nM T00407 CMF86O 137348600 IC50 = 24000 nM T00407 CW1IF3 137348845 IC50 = 22000 nM T00407 C4VNB8 137369426 IC50 = 45 nM T00407 CTM7U5 137628634 IC50 = 45 nM T00407 CS6U7Y 137631402 IC50 = 720 nM T00407 C53KAO 137631500 IC50 = 4900 nM T00407 CU49YR 137631543 IC50 > 10000 nM T00407 COP3H7 137631627 IC50 = 120 nM T00407 CA2VS4 137631629 IC50 = 3900 nM T00407 C0Y3UF 137631784 IC50 = 10100 nM T00407 CNZS84 137631821 IC50 > 10000 nM T00407 CUE7F1 137631875 IC50 = 490 nM T00407 CR5FO2 137632087 Ki > 40000 nM T00407 C25OZB 137632559 IC50 > 20000 nM T00407 C7F4MJ 137632577 Ki = 190 nM T00407 CA2D8W 137632690 Ki > 40000 nM T00407 C5JP8O 137633986 IC50 = 12 nM T00407 CF9I7B 137634124 IC50 = 170 nM T00407 CYU6T2 137634563 IC50 > 20000 nM T00407 CX9OI0 137634784 IC50 = 180 nM T00407 C9XVL1 137635109 IC50 = 11200 nM T00407 CS27YB 137635150 IC50 = 401 nM T00407 CM9P2A 137635443 IC50 = 2300 nM T00407 CQW04U 137635588 Ki = 8.7 nM T00407 CBX4I3 137635735 IC50 = 530 nM T00407 C0D1LR 137635790 IC50 > 20000 nM T00407 CO0UN6 137635792 IC50 = 1500 nM T00407 CWYU04 137635881 IC50 > 10000 nM T00407 C2P8AM 137636088 Ki = 9 nM T00407 CQT3A9 137636309 IC50 > 100000 nM T00407 CYZJ80 137636683 IC50 = 4900 nM T00407 CO08EU 137636712 Ki = 2500 nM T00407 CCAP49 137636933 IC50 > 20000 nM T00407 C92AIX 137637032 Ki = 26 nM T00407 C69BGA 137637084 IC50 = 2470 nM T00407 C7NZ4E 137637179 IC50 = 3200 nM T00407 C05CVD 137637565 IC50 = 520 nM T00407 C1AB7Q 137637710 IC50 > 10000 nM T00407 CT2D8X 137638314 IC50 = 13000 nM T00407 CRN21V 137638824 IC50 = 1500 nM T00407 CVK32T 137639306 Ki = 160 nM T00407 C6ZG0E 137639443 IC50 = 160 nM T00407 CP2HK4 137639600 IC50 = 3800 nM T00407 CV1EP8 137639742 IC50 = 37000 nM T00407 CFS67E 137640120 IC50 = 1810 nM T00407 C5MS7I 137640141 IC50 = 40 nM T00407 CKUX65 137640422 IC50 = 6400 nM T00407 CF42ZW 137640560 IC50 = 8590 nM T00407 CJG6R8 137640750 IC50 = 3400 nM T00407 C0SYB2 137640929 IC50 = 18400 nM T00407 CL4FK6 137641456 IC50 > 20000 nM T00407 COK20S 137641504 IC50 = 1400 nM T00407 CXH59O 137641530 IC50 > 10000 nM T00407 C01BVT 137642411 IC50 = 2000 nM T00407 CMX9U6 137642634 IC50 > 10000 nM T00407 COY3A6 137642659 IC50 = 9200 nM T00407 C9XZ3O 137643020 IC50 = 2700 nM T00407 CGE1L2 137643245 Ki = 430 nM T00407 C41QFV 137643280 IC50 > 10000 nM T00407 C36RVQ 137643517 IC50 > 10000 nM T00407 CP28JU 137643679 IC50 > 10000 nM T00407 CD8VQ1 137643820 Ki > 40000 nM T00407 CDK90I 137643908 IC50 < 50 nM T00407 CQ0YM6 137643978 IC50 = 2200 nM T00407 CZXP42 137644405 IC50 > 20000 nM T00407 CRJ2W3 137644677 IC50 = 630 nM T00407 C2T8WQ 137644823 IC50 = 18500 nM T00407 C7G3SF 137644942 IC50 = 640 nM T00407 CYBP84 137644977 IC50 = 200 nM T00407 C37MBU 137645618 IC50 > 10000 nM T00407 CTG91Q 137646067 IC50 = 320 nM T00407 C0R3FG 137646519 IC50 = 4200 nM T00407 CGQ3X2 137647012 IC50 = 68 nM T00407 CWJ7N5 137647079 IC50 = 6900 nM T00407 CJ9UI7 137647118 IC50 > 20000 nM T00407 CXD50J 137647775 IC50 = 16800 nM T00407 CGX65O 137647885 IC50 > 20000 nM T00407 C2HTJ9 137648078 IC50 = 180 nM T00407 C8QO2D 137648257 Ki = 110 nM T00407 C6AXY7 137648298 IC50 = 17 nM T00407 CK16RO 137648883 IC50 = 5700 nM T00407 CV3J1C 137648959 IC50 > 10000 nM T00407 C9TC6G 137648962 Ki = 4.4 nM T00407 C0NR8F 137649215 IC50 = 130 nM T00407 C89VWP 137649346 IC50 = 6000 nM T00407 CQ9G8P 137649425 IC50 > 10000 nM T00407 CC2V9L 137649517 IC50 < 5 nM T00407 CA0G8B 137649726 IC50 < 50 nM T00407 C85QNS 137649815 IC50 = 9400 nM T00407 CKN60B 137649822 IC50 > 120000 nM T00407 CO7K6Y 137649906 IC50 = 13200 nM T00407 CZ4VH1 137650214 IC50 = 17 nM T00407 CM6S0X 137650255 IC50 > 20000 nM T00407 CQ5WF3 137650342 IC50 = 225 nM T00407 CM1WG7 137650502 IC50 = 3.1 nM T00407 CC34KQ 137650533 IC50 = 4600 nM T00407 CLGI76 137650651 IC50 > 10000 nM T00407 C4Y8HV 137650663 IC50 = 4600 nM T00407 C52APO 137650788 IC50 = 1530 nM T00407 C6FXI4 137650878 IC50 = 6370 nM T00407 CY0G4J 137650944 IC50 = 1040 nM T00407 CE42GP 137650954 IC50 = 4100 nM T00407 CSV15U 137650957 IC50 = 52000 nM T00407 C8UT7D 137651043 Ki = 460 nM T00407 C1MA2K 137651137 IC50 > 20000 nM T00407 CV9F6J 137651164 IC50 > 120000 nM T00407 C5Y0DH 137651263 IC50 > 20000 nM T00407 C2SMF1 137651591 Ki = 370 nM T00407 C6SKI2 137651884 IC50 > 20000 nM T00407 CHN7A8 137652035 IC50 = 4500 nM T00407 CMYI27 137652124 IC50 = 7400 nM T00407 CG9OR2 137652284 IC50 > 10000 nM T00407 C82CEA 137652287 IC50 = 36 nM T00407 CB3J9E 137652309 IC50 = 25000 nM T00407 C5ANC9 137652708 IC50 = 430 nM T00407 CCZD32 137652808 IC50 = 9400 nM T00407 CT17HB 137653121 Ki = 2200 nM T00407 CHU2W4 137653154 IC50 > 120000 nM T00407 CM9HL5 137653223 IC50 = 140 nM T00407 CA4WO8 137653484 Ki = 140 nM T00407 C7Y6IH 137653562 IC50 = 4300 nM T00407 C7APB1 137653732 IC50 = 3240 nM T00407 CL1V9T 137654008 IC50 = 4400 nM T00407 C7G8AR 137654107 IC50 = 490 nM T00407 CZ1K6N 137654718 Ki = 10000 nM T00407 C3OX9R 137655043 IC50 > 10000 nM T00407 C7L6MV 137655172 IC50 > 20000 nM T00407 CVH74T 137655200 Ki = 1200 nM T00407 CWPO58 137655523 IC50 = 1040 nM T00407 CGC79R 137655670 IC50 > 10000 nM T00407 CQ9UL6 137655871 IC50 = 390 nM T00407 CM7Y4D 137655923 IC50 = 13900 nM T00407 C5B7LO 137656022 IC50 = 5800 nM T00407 CX35DY 137656164 IC50 = 8300 nM T00407 C8BP5R 137656667 IC50 = 15000 nM T00407 C1SBT0 137656977 IC50 > 10000 nM T00407 CW9C8L 137657087 IC50 = 14400 nM T00407 C1YOL6 137657448 Ki = 100 nM T00407 C5TEY3 137657620 IC50 > 80000 nM T00407 C9LHE3 137657639 IC50 > 10000 nM T00407 C9DGJ2 137657716 Ki = 8.2 nM T00407 C1N7LY 137658279 IC50 > 20000 nM T00407 CE3CQ5 137659158 IC50 = 1600 nM T00407 CAS5V7 137659228 Ki = 3.4 nM T00407 C5TDP8 137660755 Ki = 3000 nM T00407 CT9Z7G 137661063 IC50 = 97 nM T00407 C7F1YH 137661082 IC50 = 9 nM T00407 CI6B7L 137661152 IC50 = 350 nM T00407 C3NPW0 137661190 IC50 = 200 nM T00407 C4XR7V 137661795 IC50 > 10000 nM T00407 C8TO4R 137662308 IC50 > 10000 nM T00407 CM3UF7 137700779 IC50 > 10000 nM T00407 CU5N8O 137701509 IC50 = 1700 nM T00407 CYV4O3 138756791 IC50 = 1300 nM T00407 CQ6XB7 139030526 IC50 = 19952.62 nM T00407 C1G9LA 139035062 Ki = 7.3 nM T00407 CPY8E7 139341516 IC50 = 10 nM T00407 COE12P 139341517 IC50 = 3600 nM T00407 C3HJI2 139341518 IC50 = 669 nM T00407 CWK82L 139341520 IC50 = 67.3 nM T00407 C3DGA7 139341522 IC50 = 11.7 nM T00407 C4CHN3 139341523 IC50 = 76 nM T00407 CRW7P5 139341524 IC50 = 9.5 nM T00407 C98TAG 139341527 IC50 = 15 nM T00407 CJ01EC 139341528 IC50 = 78.6 nM T00407 C5F7OS 139341530 IC50 > 1000 nM T00407 COY2D4 139341532 IC50 = 128 nM T00407 CVLH98 139341533 IC50 = 1600 nM T00407 C6BV5E 139341541 IC50 = 4.2 nM T00407 CWM81B 139341544 IC50 = 4.7 nM T00407 CF1VL4 139341553 IC50 = 117 nM T00407 CF8LU1 139341570 IC50 = 16.2 nM T00407 C3SVA5 139341572 IC50 = 3.5 nM T00407 CL9XU2 139341575 IC50 = 28.4 nM T00407 C69JHS 139341584 IC50 = 229 nM T00407 CJ9TL3 139341588 IC50 > 2000 nM T00407 C7IN1U 139341589 IC50 = 438 nM T00407 C0HT4J 139341591 IC50 = 97.9 nM T00407 CF2D6W 139341726 IC50 = 788 nM T00407 CI1H2T 139341727 IC50 = 740 nM T00407 C9K8YX 139341747 IC50 > 1000 nM T00407 C4YMW6 139341818 IC50 = 71.3 nM T00407 CYQ79A 139382567 IC50 > 20000 nM T00407 C24DCX 139547911 IC50 = 296 nM T00407 C0D6ZN 141531706 IC50 > 100 nM T00407 C1YV7C 141531707 IC50 > 100 nM T00407 C8ZQ2U 141736359 IC50 > 20000 nM T00407 C5VNM4 141736367 IC50 > 20000 nM T00407 C4H6ZE 141759312 IC50 = 930 nM T00407 CH0I8X 142296514 IC50 = 238.5 nM T00407 CR2UQ8 142296515 IC50 = 20.4 nM T00407 CDK17C 142296518 IC50 = 1470 nM T00407 C9U5OC 142296519 IC50 = 1350 nM T00407 C45FBX 142296520 IC50 = 350 nM T00407 CV01UW 142296521 IC50 = 54.6 nM T00407 C9F8QZ 142296524 IC50 = 125.5 nM T00407 C4B7JP 142296525 IC50 = 10.3 nM T00407 C12UVJ 142296527 IC50 = 1030 nM T00407 CAI65C 142296528 IC50 > 1000 nM T00407 CL56YI 142296532 IC50 = 730 nM T00407 C8I1XZ 142296533 IC50 = 10.5 nM T00407 C6BL0T 142296538 IC50 = 389 nM T00407 CB17LA 142296539 IC50 = 770 nM T00407 CJLX96 142296540 IC50 = 17.2 nM T00407 CNTR63 142296543 IC50 = 124.5 nM T00407 CCI89P 142296544 IC50 > 1000 nM T00407 C0AZR5 142296546 IC50 = 20.9 nM T00407 CH1DE5 142296549 IC50 = 320 nM T00407 CJGR35 142296552 IC50 = 22.3 nM T00407 C1O4EU 142296553 IC50 = 189.5 nM T00407 C8JD1T 142296555 IC50 = 31.3 nM T00407 CW5UI4 142296557 IC50 = 81.7 nM T00407 C9BGH7 142296560 IC50 = 73.8 nM T00407 CKR85F 142296562 IC50 = 62.3 nM T00407 CH5Q3R 142296563 IC50 = 175.8 nM T00407 C1IX7Q 142296567 IC50 = 46.4 nM T00407 C26QKE 142296568 IC50 = 1574.5 nM T00407 CU2FS3 142296570 IC50 = 27.4 nM T00407 CQV3X9 142296573 IC50 = 17.4 nM T00407 CT7NJ3 142296575 IC50 = 60.7 nM T00407 CH9UR4 142296576 IC50 = 760 nM T00407 CD8ZU4 142296577 IC50 = 380 nM T00407 C6VJQ4 142296579 IC50 = 199 nM T00407 C6N2KD 142296581 IC50 = 36.2 nM T00407 CM8D2W 142296582 IC50 = 20.2 nM T00407 C29URB 142296583 IC50 = 770 nM T00407 C7O2GC 142296584 IC50 = 1040 nM T00407 C9R8DG 142296585 IC50 = 357 nM T00407 CM51HE 142296589 IC50 = 13.6 nM T00407 CPC79Y 142296592 IC50 = 37.9 nM T00407 CX1F8A 142296595 IC50 = 10.6 nM T00407 CVZ0W4 142296596 IC50 = 270 nM T00407 CI73SX 142296601 IC50 = 285.5 nM T00407 C7VS9Z 142296602 IC50 = 250 nM T00407 CP2M0O 142296603 IC50 = 240 nM T00407 CW1FX5 142296604 IC50 = 177.5 nM T00407 CZSB40 142296605 IC50 = 152.5 nM T00407 CJAM56 142296607 IC50 = 15.9 nM T00407 CIWV81 142296611 IC50 = 1530 nM T00407 CG6X3A 142535938 EC50 = 526 nM T00407 CQB16E 142577810 IC50 = 398.11 nM T00407 CWYC72 142577823 IC50 = 398.11 nM T00407 CM3R1C 142577824 IC50 = 630.96 nM T00407 C6E2DB 142577846 IC50 = 316.23 nM T00407 C6X5VA 142577862 IC50 = 501.19 nM T00407 CWV83D 142577883 IC50 = 1258.93 nM T00407 C6YPL1 142740580 IC50 = 25.12 nM T00407 CWE84Z 142740586 IC50 = 39.81 nM T00407 CWHP86 142740595 IC50 = 79.43 nM T00407 C0WX3V 145829181 IC50 = 100 nM T00407 CXV80B 145829182 IC50 = 2479 nM T00407 CD6U7X 145925666 IC50 = 87.7 nM T00407 C8OD1K 145925690 IC50 = 165.96 nM T00407 C7EB9S 145945981 IC50 = 4.5 nM T00407 CR6V5X 145946095 IC50 = 12589.25 nM T00407 C0CE9F 145946096 IC50 = 6309.57 nM T00407 C25ZQV 145946097 IC50 = 251.19 nM T00407 C6VNJ7 145949319 IC50 = 510 nM T00407 CZ9U2C 145949385 IC50 = 270 nM T00407 C1CIP3 145949560 IC50 = 530 nM T00407 CS96DV 145950283 IC50 = 2120 nM T00407 C48MVS 145950376 IC50 = 2270 nM T00407 C1VM4D 145950404 IC50 = 18720 nM T00407 CUTA34 145950411 IC50 = 180 nM T00407 CH93SO 145950673 IC50 = 13300 nM T00407 CW58CR 145950888 IC50 = 610 nM T00407 C96NCH 145950955 IC50 > 20000 nM T00407 C21NAZ 145951567 IC50 = 170 nM T00407 C1XZG5 145951828 IC50 = 280 nM T00407 C1HLK5 145951928 IC50 = 17 nM T00407 CEA0I1 145952035 IC50 = 69230 nM T00407 C3ZV1O 145952497 IC50 > 20000 nM T00407 CRL42T 145953028 IC50 = 580 nM T00407 CNU28F 145953072 IC50 = 23060 nM T00407 C9I0SC 145953078 IC50 = 830 nM T00407 CVN8A5 145953287 IC50 = 620 nM T00407 CI9U2L 145953592 IC50 = 490 nM T00407 CC5D1Q 145953654 IC50 = 1330 nM T00407 CSR9N7 145953663 IC50 = 480 nM T00407 CBNI84 145953835 IC50 = 1170 nM T00407 C0ZTC4 145954129 IC50 = 110 nM T00407 C2MYA1 145954210 IC50 = 790 nM T00407 CTE74G 145954441 IC50 > 20000 nM T00407 CH14TJ 145954453 IC50 = 860 nM T00407 CBYF17 145954698 IC50 = 290 nM T00407 CR6OX1 145954766 IC50 = 120 nM T00407 CMCH58 145954903 IC50 = 13260 nM T00407 C6D0OT 145955789 IC50 > 20000 nM T00407 CMQ3J7 145955860 IC50 = 4250 nM T00407 CF0EK4 145956136 IC50 = 230 nM T00407 CB61VZ 145956237 IC50 = 270 nM T00407 C8M5DP 145956320 IC50 = 200 nM T00407 C8SC9E 145956329 IC50 = 3540 nM T00407 CIU29S 145956336 IC50 = 1140 nM T00407 CCNU52 145956492 IC50 = 570 nM T00407 C50CSO 145956910 IC50 = 180 nM T00407 CN5YO3 145957310 IC50 > 20000 nM T00407 CEJA84 145957398 IC50 = 50750 nM T00407 C9J2GS 145957453 IC50 > 20000 nM T00407 C42KZE 145957509 IC50 = 400 nM T00407 CIW97K 145957788 IC50 = 270 nM T00407 CSK9W5 145957886 IC50 = 520 nM T00407 CX7C4V 145958221 IC50 = 3640 nM T00407 CIDU52 145958263 IC50 = 340 nM T00407 C0IN8H 145958454 IC50 = 460 nM T00407 C7C5WL 145958595 IC50 = 2190 nM T00407 C2VNR7 145958596 IC50 = 290 nM T00407 C0CUF6 145958773 IC50 = 1170 nM T00407 CA9UQ0 145959024 IC50 > 1000 nM T00407 CT96GS 145959255 IC50 = 410 nM T00407 C30DFL 145959472 IC50 = 27520 nM T00407 CDNG83 145959505 IC50 = 150 nM T00407 C8AP9H 145959530 IC50 = 360 nM T00407 CIZW13 145959848 IC50 = 1430 nM T00407 C85NDV 145959886 IC50 = 6070 nM T00407 CGA86D 145960246 IC50 = 12710 nM T00407 C5R2OX 145960489 IC50 = 602.56 nM T00407 CR7Q6O 145960620 IC50 = 1230.27 nM T00407 C8DIH1 145960623 IC50 = 1100 nM T00407 CRPN57 145960718 IC50 = 585 nM T00407 CBC6Z8 145960723 IC50 = 2238.72 nM T00407 CG27BX 145961203 IC50 = 120 nM T00407 CL4XG1 145961395 IC50 = 793 nM T00407 CSDU51 145961590 IC50 = 842 nM T00407 CDZ8R4 145961700 IC50 = 722 nM T00407 CY2B3F 145961967 IC50 = 630.96 nM T00407 C90WEP 145961969 IC50 = 4680 nM T00407 C5PN9T 145962081 IC50 = 810 nM T00407 CJY05H 145962174 IC50 = 165.96 nM T00407 CKQ3G4 145962258 IC50 = 1412.54 nM T00407 CAF0K5 145962473 IC50 = 269.15 nM T00407 CEZ30H 145962475 IC50 = 4265.8 nM T00407 C49WON 145962542 IC50 = 489.78 nM T00407 C5T0KG 145962602 IC50 = 945 nM T00407 CBU2O7 145962767 IC50 = 478 nM T00407 C3YL0V 145962799 IC50 = 302 nM T00407 C6V3LN 145962814 IC50 = 3800 nM T00407 CMW3L6 145963581 IC50 = 380.19 nM T00407 CM4RN5 145963629 IC50 = 954.99 nM T00407 CH4QA2 145963723 IC50 = 3235.94 nM T00407 CC06PY 145963915 IC50 = 41900 nM T00407 CT3G0N 145963947 IC50 = 630.96 nM T00407 CU7WE5 145964377 Ki = 6.5 nM T00407 CC17DU 145964393 IC50 = 253 nM T00407 CH06LF 145964543 IC50 = 104 nM T00407 CT28NG 145964553 IC50 = 316.23 nM T00407 C4CIF7 145965008 IC50 = 794.33 nM T00407 C6EOB0 145965052 IC50 = 184.5 nM T00407 C72YHJ 145965062 Ki = 57 nM T00407 CD2WO6 145965211 IC50 = 5011.87 nM T00407 CCW5X8 145965219 IC50 = 107 nM T00407 C3FJ0L 145965372 IC50 = 100 nM T00407 CKNE25 145965382 IC50 = 251.19 nM T00407 C6M3FN 145965388 Ki = 17 nM T00407 CJ07ZP 145965402 IC50 = 125.89 nM T00407 C0X8PE 145965751 IC50 = 1000 nM T00407 CQC15M 145966021 IC50 = 79.43 nM T00407 CCTY08 145966026 IC50 = 107.5 nM T00407 C2Q7ES 145966038 IC50 = 100 nM T00407 CJ27UK 145966193 Ki < 0.5 nM T00407 CJ5BC4 145966522 IC50 = 2.3 nM T00407 C4ED6N 145966560 IC50 = 501.19 nM T00407 CE4D5F 145966579 IC50 = 596 nM T00407 C8XR2B 145966639 IC50 = 25118.86 nM T00407 C5BFX2 145966845 IC50 = 2511.89 nM T00407 CC05ZI 145967006 IC50 = 316.23 nM T00407 C4Y0PN 145967100 IC50 > 20000 nM T00407 C0T3BJ 145967243 IC50 = 1000 nM T00407 CYV74C 145967245 Ki = 10.5 nM T00407 C1V2DR 145967422 IC50 = 50.12 nM T00407 CHQ9L0 145967434 IC50 = 168 nM T00407 C2M7TI 145967443 IC50 = 370 nM T00407 CXWZ04 145967512 IC50 = 421 nM T00407 CX1C4W 145967999 IC50 = 4.3 nM T00407 CV4LN0 145968329 IC50 = 72000 nM T00407 C7SC5G 145968551 IC50 = 121000 nM T00407 CT06PA 145969741 IC50 = 15000 nM T00407 C9S8GB 145969777 IC50 > 200000 nM T00407 C0ZN2W 145969902 IC50 = 26000 nM T00407 C4YE5O 145970005 IC50 = 49000 nM T00407 CS6N3Y 145970287 IC50 > 10000 nM T00407 C13UOX 145970508 IC50 = 158.49 nM T00407 CO4RB3 145970920 IC50 = 24000 nM T00407 C7SK4T 145971247 IC50 > 1000 nM T00407 CDB65R 145971415 IC50 = 125.89 nM T00407 CCAT53 145971461 IC50 = 200 nM T00407 CF37MT 145971516 IC50 = 210 nM T00407 C3BSE8 145971523 IC50 = 590 nM T00407 C4GX3P 145971629 IC50 = 630.96 nM T00407 C9Q5RW 145971747 IC50 = 880 nM T00407 CV0TS2 145971844 IC50 = 794.33 nM T00407 CH8Y6A 145971920 IC50 = 1020 nM T00407 CIJO67 145972096 IC50 = 650 nM T00407 CV83ED 145972103 Ki = 1.2 nM T00407 C4D8RC 145972215 IC50 = 100 nM T00407 C0PFQ7 145972286 IC50 > 10000 nM T00407 CN70KV 145972360 IC50 = 95 nM T00407 CNU4O9 145972623 IC50 = 5100 nM T00407 C2RTO8 145972845 IC50 = 107 nM T00407 CQ35BN 145972969 IC50 = 1258.93 nM T00407 CD4A3Y 145973334 IC50 > 20000 nM T00407 C1Z3WQ 145973981 IC50 = 794.33 nM T00407 CWQ6A5 145974124 Ki = 2.7 nM T00407 CP49HN 145974181 IC50 > 20000 nM T00407 CXF6B5 145974721 IC50 = 501.19 nM T00407 CW37DI 145974796 IC50 = 87 nM T00407 CE7O2Z 145974859 Ki < 0.5 nM T00407 CG0D7U 145974979 IC50 = 100 nM T00407 CA85TK 145975493 IC50 > 20000 nM T00407 C6R2YM 145975649 IC50 = 2579 nM T00407 CTAZ41 145975701 IC50 > 50000 nM T00407 CW56PH 145975703 IC50 = 28 nM T00407 CRZ78W 145975795 IC50 = 630.96 nM T00407 CH57GW 145975937 IC50 = 186 nM T00407 CN4O0K 145976012 IC50 = 310 nM T00407 CKG83I 145976334 Ki = 641 nM T00407 CG0ZO6 145976380 IC50 = 794.33 nM T00407 CAL91V 145976398 IC50 = 158.49 nM T00407 CS05DX 145976415 IC50 = 1584.89 nM T00407 CR28YS 145976646 IC50 = 59 nM T00407 C26XFE 145976805 IC50 = 158.49 nM T00407 C1F7DT 145976814 IC50 = 398.11 nM T00407 C7J1IZ 145976831 IC50 = 168 nM T00407 CVJ61U 145977109 IC50 = 690 nM T00407 C3NUY9 145977309 Ki = 2.7 nM T00407 COD4I9 145977320 IC50 = 199.53 nM T00407 CG5TD0 145977365 IC50 = 63.1 nM T00407 C6M2CY 145977402 IC50 = 1258.93 nM T00407 CX13RH 145977417 IC50 = 1258.93 nM T00407 C63KPH 145977495 IC50 = 630.96 nM T00407 CB9F1X 145977980 IC50 = 94 nM T00407 C0MD9U 145978238 IC50 = 183 nM T00407 CJE53V 145978248 Ki = 7.7 nM T00407 C6S9BA 145978560 IC50 = 501.19 nM T00407 CSKC69 145978686 IC50 = 794.33 nM T00407 C8CO6S 145978782 IC50 = 50.12 nM T00407 C3LC2N 145978789 Ki = 4.4 nM T00407 CK4PH5 145978839 IC50 = 1108.5 nM T00407 CXC9E4 145978854 IC50 = 63.1 nM T00407 C0AI4C 145979130 IC50 = 25430 nM T00407 CAV7J5 145979375 IC50 = 1440 nM T00407 CV4TW9 145979405 IC50 = 6 nM T00407 CY6S4Z 145979516 IC50 = 4790 nM T00407 CYZ14K 145979939 IC50 = 12010 nM T00407 CHM8L7 145981045 IC50 = 1995.26 nM T00407 C9AUV1 145981148 IC50 = 630.96 nM T00407 CVYU19 145981267 IC50 = 2960 nM T00407 CJ0T1R 145981696 IC50 = 3870 nM T00407 CRXH81 145981836 IC50 = 794.33 nM T00407 CI5H7L 145982424 IC50 = 4730 nM T00407 CJ3FL8 145982835 IC50 > 50118.72 nM T00407 CA2W8M 145984295 IC50 = 31622.78 nM T00407 C4HWL1 145984406 IC50 = 40100 nM T00407 CE05ZV 145984432 IC50 = 25118.86 nM T00407 CV4GH7 145984467 IC50 = 7943.28 nM T00407 CT6V0I 145985751 IC50 = 6309.57 nM T00407 C0GHY5 145986052 IC50 = 158489.32 nM T00407 C69GXS 145986370 IC50 = 25118.86 nM T00407 C3OS2V 145987227 IC50 > 50000 nM T00407 C3QEX7 145987948 IC50 = 81000 nM T00407 CK20BY 145988169 Ki = 152 nM T00407 CY0OK3 145988346 IC50 = 794.33 nM T00407 CHL20Z 145988638 IC50 > 50000 nM T00407 COZ5J9 145989122 IC50 = 5011.87 nM T00407 COC35Q 145989187 IC50 = 501.19 nM T00407 CN4HR9 145989400 IC50 = 4770 nM T00407 CKP14Z 145989459 IC50 > 50000 nM T00407 C0NHS8 145989546 IC50 > 50000 nM T00407 CGY12F 145989646 IC50 = 2730 nM T00407 C7WRS3 145989682 IC50 = 2 nM T00407 CC9OS3 145989699 IC50 = 630.96 nM T00407 CC6NH9 145989855 IC50 = 1584.89 nM T00407 CSF47C 145990617 IC50 = 9320 nM T00407 CM5N9Y 145991689 IC50 = 1000 nM T00407 CSG40R 145991750 IC50 > 50000 nM T00407 C1SQD3 145992400 IC50 = 3590 nM T00407 CSN3C8 145992593 IC50 = 501.19 nM T00407 C1DP4O 146027046 Ki = 1.1 nM T00407 CK98QJ 146035912 IC50 > 50118.72 nM T00407 C53GZM 146037608 IC50 = 130 nM T00407 CZY8D7 146037609 IC50 = 2700 nM T00407 CL9TB0 146037610 IC50 > 10000 nM T00407 CBRE71 146047136 IC50 = 2.6 nM T00407 C3XOR2 146322224 IC50 = 6.1 nM T00407 C9TW5Q 146322225 IC50 = 100.4 nM T00407 CR12JW 146322226 IC50 = 7.9 nM T00407 CGV47C 146322227 IC50 = 9.6 nM T00407 CAE39T 146322229 IC50 = 8.7 nM T00407 CZ5KA1 146322241 IC50 = 142 nM T00407 CI2HL1 146322248 IC50 = 5.2 nM T00407 CQF42T 146322251 IC50 = 9.4 nM T00407 CH1I3X 146322264 IC50 = 4.2 nM T00407 C8LXY6 146322265 IC50 = 8.6 nM T00407 C3MT7G 146322268 IC50 = 5.9 nM T00407 C3R5OK 146322269 IC50 = 4.6 nM T00407 CJO2X3 146322270 IC50 = 5.3 nM T00407 CQ0S8V 146322271 IC50 = 7 nM T00407 CQG82Z 146322272 IC50 = 4.8 nM T00407 CC6RE8 146322280 IC50 = 4.6 nM T00407 C1G3IC 146322281 IC50 = 6.6 nM T00407 CFV96I 146322282 IC50 = 27.2 nM T00407 C4WYD7 146322283 IC50 = 6.8 nM T00407 C3QPV4 146322290 IC50 = 5.4 nM T00407 CG50HD 146322292 IC50 = 7.1 nM T00407 C2XWK6 146322293 IC50 = 5.8 nM T00407 CT6XO0 146322294 IC50 = 5.7 nM T00407 CZ3T7Q 146322295 IC50 = 14.4 nM T00407 C2ZVK5 146322296 IC50 = 9.5 nM T00407 CLK37M 147133615 Ki = 54.4 nM T00407 CTQ01S 147823626 Ki = 736 nM T00407 COU42L 147881243 IC50 = 92 nM T00407 CGW0K7 148225107 Ki = 376 nM T00407 CPQ57V 148251486 IC50 = 39.6 nM T00407 C5O7VJ 148648403 Ki = 50.3 nM T00407 CIUR70 149201098 Ki = 102 nM T00407 CWG10H 151364732 IC50 = 1190 nM T00407 CP5V2U 152625752 IC50 = 9.7 nM T00407 C6I7OZ 152636346 IC50 = 980 nM T00407 C7LM4U 153534003 IC50 = 1930 nM T00407 CP1V9H 153534004 IC50 = 1770 nM T00407 C9FIY4 153534005 IC50 = 710 nM T00407 CVT63S 153534008 IC50 = 2190 nM T00407 CZCD51 155352257 IC50 = 3900 nM T00407 CM4V9L 155352262 IC50 = 11000 nM T00407 C40KOR 155352277 IC50 > 100000 nM T00407 CZ50CJ 155352280 IC50 = 4500 nM T00407 C5K3FL 155352284 IC50 > 100000 nM T00407 CG6HY5 155352290 IC50 > 100000 nM T00407 C1ZFB8 155352296 IC50 > 100000 nM T00407 CPZ64D 155352301 IC50 = 1700 nM T00407 CB8EF6 155352304 IC50 = 61000 nM T00407 C02EIO 155352320 IC50 > 100000 nM T00407 C40RYV 155352344 IC50 > 100000 nM T00407 CHG13B 155352345 IC50 = 9700 nM T00407 CFD6H1 155352361 IC50 = 75000 nM T00407 CL2ZE0 155352369 IC50 > 100000 nM T00407 C8GZL5 155352384 IC50 = 1300 nM T00407 CFK2B1 155352401 IC50 = 102000 nM T00407 C0RO5V 155352412 IC50 = 12000 nM T00407 CZ1A8M 155352425 IC50 = 97000 nM T00407 C7U0VB 155352430 IC50 = 27000 nM T00407 C9FR3V 155510506 IC50 = 5930 nM T00407 CPY92M 155510533 IC50 = 310 nM T00407 CLMX96 155510847 Ki = 1 nM T00407 C2CD3Y 155510879 IC50 = 5540 nM T00407 CQUC76 155510893 Ki = 92 nM T00407 C98HOQ 155511096 Ki = 0.5 nM T00407 C9AXU3 155511227 IC50 = 169.1 nM T00407 CI6SA1 155511268 Ki = 945 nM T00407 CO0B1A 155511836 IC50 = 1529 nM T00407 C3R1EO 155511887 Ki = 15.85 nM T00407 C0LH8C 155511921 IC50 > 10000 nM T00407 C2D1SB 155512075 IC50 = 10000 nM T00407 CT2H3S 155512097 IC50 = 3100 nM T00407 CF6S3U 155512187 IC50 = 223 nM T00407 CD3LA9 155512613 IC50 > 50118.72 nM T00407 C51DIZ 155512733 IC50 = 62 nM T00407 C76QMK 155513141 Ki = 14.8 nM T00407 C5WUJ6 155513192 IC50 > 10000 nM T00407 C1D6MT 155513275 Ki = 50.12 nM T00407 CNQ9S2 155513363 IC50 = 205.2 nM T00407 CG47KU 155513649 Ki = 20 nM T00407 C9IUC2 155513805 IC50 = 1790 nM T00407 CF0GQ6 155513971 IC50 = 501.19 nM T00407 CP6VY4 155514289 Ki = 13 nM T00407 CI5CW6 155514299 Ki = 3.2 nM T00407 CS65YK 155514303 IC50 = 10 nM T00407 CH9KM8 155514491 IC50 = 655.8 nM T00407 C5JMW2 155514540 IC50 = 68 nM T00407 CNSC23 155514584 IC50 = 10 nM T00407 C30COX 155514594 IC50 = 6300 nM T00407 C27LFN 155514936 IC50 = 560 nM T00407 CX5W9H 155515117 IC50 = 5000 nM T00407 CE13CA 155515130 IC50 > 50118.72 nM T00407 C4THO2 155515131 Ki = 9.6 nM T00407 CH0LR3 155515173 IC50 = 50 nM T00407 CZU79I 155515498 IC50 = 6740 nM T00407 C8NC6V 155515565 IC50 = 8 nM T00407 C4GEL0 155515650 Ki = 18 nM T00407 CT03IV 155516089 IC50 = 1569 nM T00407 CZYP31 155516103 Ki = 1.3 nM T00407 C2GB7R 155516112 IC50 = 54 nM T00407 CPM43N 155516232 IC50 > 50118.72 nM T00407 CTI9Q6 155516388 IC50 = 19006 nM T00407 CNCH70 155516682 Ki = 1.1 nM T00407 CX6N4Z 155516719 IC50 = 1584.89 nM T00407 CDCH75 155516938 IC50 = 2598 nM T00407 CT5ZC6 155516968 IC50 = 22 nM T00407 C23BXS 155517049 IC50 > 50118.72 nM T00407 CP3K4R 155517232 IC50 = 44 nM T00407 CF0C7V 155517447 IC50 = 20.9 nM T00407 CS28LW 155517521 Ki = 47.3 nM T00407 CE0CX6 155517720 IC50 = 3466 nM T00407 C6Q3JK 155517968 IC50 > 50118.72 nM T00407 C8HK5X 155518008 IC50 = 1000 nM T00407 C32FEU 155518033 IC50 = 163.7 nM T00407 CFP24B 155518498 IC50 = 15848.93 nM T00407 CGBZ95 155518530 IC50 = 17.4 nM T00407 CBM34J 155518876 Ki = 3.162 nM T00407 CP2T0H 155519067 Ki = 413 nM T00407 C2GN1Y 155519159 IC50 = 5600 nM T00407 CHP0T5 155519310 IC50 = 10 nM T00407 C5KZG7 155519527 IC50 = 73 nM T00407 CW4HJ7 155519805 IC50 = 12.6 nM T00407 C8NL9U 155519897 IC50 = 140 nM T00407 CFVU05 155519921 IC50 = 480 nM T00407 C1JT3F 155520065 IC50 = 91.3 nM T00407 CY0A8O 155520236 IC50 = 167.1 nM T00407 CMVW63 155520501 IC50 = 37 nM T00407 C95RHU 155520664 IC50 = 1500 nM T00407 CGUX31 155520762 IC50 = 6680 nM T00407 CSPY94 155520847 Ki = 1.8 nM T00407 CB49NL 155521254 IC50 = 12589.25 nM T00407 C7UKD6 155521295 Ki = 617 nM T00407 C5F1JC 155521775 IC50 = 6020 nM T00407 CC30UG 155521851 IC50 > 50118.72 nM T00407 CAL9J8 155521991 IC50 = 1130 nM T00407 CH14KR 155522315 IC50 = 6000 nM T00407 CP9VQ4 155522638 Ki = 15 nM T00407 C0SE4F 155522830 Ki = 3.7 nM T00407 C0AP3M 155522854 IC50 < 1.995 nM T00407 C30NMB 155523002 IC50 = 1645 nM T00407 CHG5N8 155523095 IC50 > 10000 nM T00407 C85RSC 155523105 Ki = 92.6 nM T00407 CH06TJ 155523190 Ki = 25 nM T00407 CJYZ12 155523212 IC50 = 205.2 nM T00407 CL1P4M 155523233 IC50 > 50118.72 nM T00407 C1LK5T 155523560 Ki = 0.7 nM T00407 C1W8JL 155523577 IC50 > 50118.72 nM T00407 C2K9NI 155523694 IC50 > 50118.72 nM T00407 C8U2FI 155523758 Ki = 0.9 nM T00407 C0VS8H 155523850 IC50 > 50118.72 nM T00407 C3NYK0 155523937 IC50 = 50118.72 nM T00407 CBPV08 155523967 IC50 = 13120 nM T00407 CB90JU 155524196 IC50 = 11400 nM T00407 C2V0OA 155524426 IC50 = 265.6 nM T00407 CXM7E8 155524802 Ki = 80.6 nM T00407 C5BX4C 155525302 IC50 = 1250 nM T00407 C7GQN6 155525350 IC50 = 251.19 nM T00407 CSN27B 155525408 Ki = 22 nM T00407 CJ0V6I 155525482 Ki = 7.943 nM T00407 CW8O7G 155525483 IC50 > 50118.72 nM T00407 CF2P9Y 155525718 IC50 = 2100 nM T00407 CH79NC 155526096 IC50 = 125.89 nM T00407 C9I2LV 155526120 IC50 = 1400 nM T00407 CO1S0P 155526228 IC50 = 22700 nM T00407 C3QV1O 155526357 Ki = 9.5 nM T00407 C6R9LD 155526395 Ki = 66 nM T00407 CRK6E2 155526401 IC50 = 794.33 nM T00407 CKD9U4 155526975 IC50 = 3200 nM T00407 CVY04U 155527380 IC50 = 13000 nM T00407 C54DZA 155527566 IC50 = 1600 nM T00407 COY9L2 155527786 IC50 = 3724 nM T00407 CK2W1L 155527824 IC50 = 36 nM T00407 C43ZEI 155527951 IC50 = 501.19 nM T00407 CV7G8W 155527989 Ki = 5.012 nM T00407 C7Y5HX 155527993 IC50 = 1810 nM T00407 CLY27Z 155528197 Ki = 1.1 nM T00407 COJ86W 155528199 Ki = 0.7 nM T00407 CX18IT 155528305 IC50 = 1696 nM T00407 CKR6V3 155528325 IC50 > 50118.72 nM T00407 C3P9LB 155528627 Ki = 63.1 nM T00407 CEVB10 155528780 IC50 = 1900 nM T00407 CV7I6Z 155528992 IC50 = 53.8 nM T00407 C7MC0H 155529162 Ki = 68.4 nM T00407 COX8K5 155529510 IC50 > 50118.72 nM T00407 CIV12T 155529744 IC50 = 9930 nM T00407 CVMC06 155529991 IC50 > 50118.72 nM T00407 CO6X5T 155530144 IC50 = 16.6 nM T00407 CL93CM 155530154 IC50 > 50118.72 nM T00407 CQ2U3P 155530217 IC50 = 299.3 nM T00407 CEI09V 155530332 IC50 = 19952.62 nM T00407 CMSW35 155530439 IC50 = 1995.26 nM T00407 C2Y1DU 155530564 IC50 = 37.5 nM T00407 CY7ST9 155530616 IC50 > 50118.72 nM T00407 CB5Z9W 155530732 IC50 = 7230 nM T00407 CEA2C7 155531097 Ki = 128 nM T00407 CNB0Z3 155531098 Ki = 0.5 nM T00407 CS48EO 155531154 IC50 = 545.2 nM T00407 CL9VB6 155531262 IC50 = 5000 nM T00407 C84UXT 155531461 IC50 = 3620 nM T00407 CV2DU3 155531469 IC50 = 2400 nM T00407 CJ93LE 155531635 IC50 = 5011.87 nM T00407 CJ3XQ0 155531658 IC50 = 63.1 nM T00407 CPY0W4 155531898 Ki = 65.4 nM T00407 COI6T9 155532041 Ki = 1.1 nM T00407 CME45L 155532169 IC50 = 1584.89 nM T00407 C7IG9L 155532175 IC50 = 47 nM T00407 CQN6G3 155532286 IC50 = 690 nM T00407 CH80JY 155532661 IC50 = 67 nM T00407 C82UPM 155532741 IC50 = 10000 nM T00407 CQ6G3D 155532785 IC50 > 10000 nM T00407 C7LUW5 155533038 IC50 = 71 nM T00407 CE3R7T 155533055 IC50 = 63 nM T00407 CQ63ZW 155533302 IC50 = 9065 nM T00407 C1HOJ8 155533481 Ki = 34.8 nM T00407 C3P5FB 155533716 IC50 = 240 nM T00407 CYL48U 155533835 IC50 = 790 nM T00407 CCS3Z2 155533896 IC50 = 630.96 nM T00407 CSDL12 155533972 Ki = 0.9 nM T00407 CY37NL 155534118 IC50 = 240 nM T00407 CRVW82 155534145 Ki = 83.7 nM T00407 CWQ9I0 155534265 IC50 = 220 nM T00407 CH39ZT 155534291 IC50 = 70 nM T00407 C9A7EM 155534450 Ki = 12.59 nM T00407 CZY5G8 155534471 IC50 = 2250 nM T00407 CFV0X3 155534492 IC50 = 81 nM T00407 CAEQ29 155534550 IC50 = 25118.86 nM T00407 C4Y2JK 155534563 Ki = 249 nM T00407 C0QV9U 155534567 IC50 = 3200 nM T00407 CWP5Z4 155534721 Ki = 0.8 nM T00407 CJUX72 155534784 IC50 = 860 nM T00407 C8R6ZI 155534867 IC50 = 8200 nM T00407 CS57MP 155535054 IC50 = 46 nM T00407 C6OP0S 155535292 Ki = 14.8 nM T00407 CBTQ04 155535301 Ki = 1.1 nM T00407 CY08SU 155535485 IC50 = 31622.78 nM T00407 C91UNV 155535585 IC50 = 2550 nM T00407 CS8XB0 155535800 IC50 = 850 nM T00407 CFM46E 155535834 IC50 = 1810 nM T00407 CG7X4Y 155536037 Ki = 12.59 nM T00407 CTYQ86 155536169 IC50 > 10000 nM T00407 C7L0ZW 155536305 IC50 = 54.8 nM T00407 C0HI7N 155536879 EC50 > 10000 nM T00407 CX01IJ 155536900 IC50 = 665.7 nM T00407 CV1FU3 155537340 IC50 = 7200 nM T00407 C02DSM 155537630 IC50 = 316.23 nM T00407 CS1KL9 155538190 IC50 = 27.5 nM T00407 CZS3A1 155538358 IC50 = 110 nM T00407 CEZJ39 155538579 IC50 = 709.4 nM T00407 C9ISB5 155538742 IC50 > 50118.72 nM T00407 CF3YQ7 155539142 IC50 = 82 nM T00407 C87NOU 155539256 IC50 = 203 nM T00407 C71XPS 155539263 Ki = 918 nM T00407 C1MQP2 155539283 IC50 = 50118.72 nM T00407 C9UP3S 155539471 IC50 = 46 nM T00407 CDCP41 155539526 IC50 = 503.2 nM T00407 C8TSQ0 155539582 IC50 = 4400 nM T00407 C7WY9X 155539828 IC50 = 113 nM T00407 CW1Z8F 155539966 Ki = 109 nM T00407 CE0FM3 155540495 IC50 = 6170 nM T00407 C62EMT 155540785 IC50 = 760 nM T00407 CV1GR7 155540862 Ki = 1.2 nM T00407 CABF92 155541119 IC50 = 750 nM T00407 C7VRN8 155541456 IC50 = 750 nM T00407 C6SG3O 155541524 IC50 = 44 nM T00407 C9SIN5 155541564 IC50 = 107 nM T00407 CXTO91 155541586 IC50 = 31622.78 nM T00407 C4UC2G 155542752 IC50 = 7300 nM T00407 CNSP97 155542781 IC50 > 50118.72 nM T00407 CF95RE 155542833 IC50 > 10000 nM T00407 CJ94RY 155543134 Ki = 17.4 nM T00407 CT8E7F 155543334 Ki = 147 nM T00407 C6FHM8 155543582 IC50 = 31622.78 nM T00407 C0IQ7Y 155544012 IC50 > 10000 nM T00407 CK2N5P 155544158 IC50 = 172.1 nM T00407 CL9Q5B 155545073 IC50 = 20 nM T00407 C2UN1K 155545446 IC50 > 10000 nM T00407 CDQ8J3 155545496 IC50 = 1600 nM T00407 C1Z6RY 155545684 Ki = 0.8 nM T00407 C1JSY3 155545907 IC50 > 10000 nM T00407 CM51BF 155546089 IC50 = 39810.72 nM T00407 CP5VY1 155546607 IC50 = 316.23 nM T00407 CH9Y8A 155546620 IC50 = 328 nM T00407 CFTR89 155546746 IC50 = 39810.72 nM T00407 CK10MI 155546815 IC50 = 48 nM T00407 C71QBN 155546897 IC50 = 550 nM T00407 CAV1O8 155546975 IC50 = 141 nM T00407 C82ZVR 155547161 Ki = 2.9 nM T00407 CUX25H 155547195 Ki = 15.9 nM T00407 CQPY75 155547500 IC50 = 5170 nM T00407 CAI8W4 155547542 IC50 = 29 nM T00407 C8ZGQ3 155547993 Ki = 174 nM T00407 CAI1K4 155548058 IC50 = 95.2 nM T00407 CNW10F 155548254 IC50 = 57 nM T00407 CST0E6 155548743 Ki = 28 nM T00407 CI12GZ 155548897 Ki = 0.5 nM T00407 CQNO46 155548910 IC50 = 31622.78 nM T00407 C8O0PK 155549061 Ki = 74.7 nM T00407 CH62AP 155549078 IC50 = 348.2 nM T00407 C4RO8G 155549970 Ki = 1.1 nM T00407 CBHN73 155550160 IC50 = 20 nM T00407 C6C3KR 155550228 IC50 = 106.7 nM T00407 CTPL52 155550409 IC50 = 540 nM T00407 C3VAJ9 155550685 IC50 = 6710 nM T00407 CNU0K9 155551427 Ki = 68 nM T00407 C1YK4R 155551595 IC50 = 708.7 nM T00407 C2VN6S 155551648 IC50 = 140 nM T00407 CJL84K 155551807 IC50 = 95 nM T00407 C4VKR0 155551851 IC50 > 50118.72 nM T00407 COG5X6 155551883 IC50 = 2410 nM T00407 CE5PB8 155551897 IC50 = 23870 nM T00407 C2FWB9 155551946 IC50 = 39810.72 nM T00407 CJ49KI 155552070 IC50 = 5920 nM T00407 C68TQG 155552169 IC50 = 260.3 nM T00407 CE6XY4 155552472 IC50 = 10 nM T00407 C5Q8NM 155552649 IC50 > 10000 nM T00407 C6SE1C 155552754 Ki = 68 nM T00407 CXB3A0 155552980 IC50 = 16341 nM T00407 C7RPH3 155553336 IC50 < 50 nM T00407 CKA2N6 155553423 Ki = 5.8 nM T00407 CHL5S0 155553610 Ki = 12.3 nM T00407 C1TLD7 155553647 IC50 = 50.12 nM T00407 CT35SU 155553650 IC50 = 39810.72 nM T00407 C4DXG8 155553846 IC50 = 3888 nM T00407 CTRE24 155554039 Ki = 0.8 nM T00407 C0VP2N 155554114 Ki = 66.2 nM T00407 CH8L1V 155554197 IC50 = 3480 nM T00407 CJN29K 155554220 IC50 = 292 nM T00407 C0SYN6 155554629 IC50 = 25118.86 nM T00407 C4UER7 155554809 IC50 = 271.2 nM T00407 CW5LG1 155554980 Ki = 284 nM T00407 CB6Q5S 155555122 IC50 = 2226 nM T00407 C7OR6T 155555165 Ki = 13 nM T00407 C1T5RH 155555385 IC50 = 61 nM T00407 CF2H3O 155555451 IC50 > 10000 nM T00407 CM7FN8 155555499 IC50 = 1170 nM T00407 CDO08V 155555578 IC50 > 50118.72 nM T00407 C12QHG 155555950 IC50 > 50118.72 nM T00407 CP2BX0 155556096 IC50 = 7943.28 nM T00407 C6JSF2 155556169 IC50 = 220 nM T00407 C83KNU 155556217 IC50 = 573.1 nM T00407 CZJ7Y4 155556283 Ki = 1.7 nM T00407 C7S8GF 155556284 IC50 > 50118.72 nM T00407 CFS7H1 155556713 IC50 = 2600 nM T00407 C5CSM3 155556861 IC50 = 1600 nM T00407 C6N1CG 155557122 IC50 > 50118.72 nM T00407 CUQ53E 155557175 IC50 = 150 nM T00407 C57UCJ 155557247 Ki = 2.1 nM T00407 C3BY7N 155557439 IC50 = 4500 nM T00407 CYM3K9 155557522 IC50 = 15848.93 nM T00407 C4I0RK 155557553 IC50 = 18500 nM T00407 C7T1PN 155557578 IC50 = 560 nM T00407 CK8O4T 155557646 IC50 > 50118.72 nM T00407 CE07MN 155557702 Ki = 68.8 nM T00407 CWHA10 155558023 IC50 > 10000 nM T00407 CM23TJ 155558268 Ki = 0.9 nM T00407 C6D4EN 155558707 IC50 = 391.3 nM T00407 C2P3TA 155558894 IC50 = 35.1 nM T00407 CSGH17 155559412 IC50 > 50118.72 nM T00407 CD4ML1 155559481 IC50 = 76 nM T00407 C5S7RE 155559494 IC50 > 10000 nM T00407 CH24ZI 155559572 IC50 = 3600 nM T00407 C2MX6K 155559855 IC50 = 158.49 nM T00407 C1C9VU 155559875 Ki = 41.5 nM T00407 CZ94JU 155560004 IC50 = 217.1 nM T00407 CSF23U 155560126 Ki = 0.6 nM T00407 C5X6EL 155560182 IC50 > 50118.72 nM T00407 CBNS45 155560213 IC50 = 155 nM T00407 C5DLU8 155560288 IC50 = 1320 nM T00407 CS1C5W 155560567 IC50 > 50118.72 nM T00407 CK45IM 155560616 Ki = 4.3 nM T00407 CI91CS 155560656 IC50 = 24000 nM T00407 C3UC7H 155560671 IC50 = 25118.86 nM T00407 C1CHQ8 155560764 Ki = 21.3 nM T00407 CG19QD 155561005 IC50 = 162 nM T00407 CI1ZU8 155561055 IC50 = 9600 nM T00407 CU2O6Z 155561457 Ki = 1.4 nM T00407 CH0Z1P 155561539 IC50 > 10000 nM T00407 CRNC43 155561660 IC50 = 1400 nM T00407 CZA5N1 155561689 EC50 = 9110 nM T00407 C3RYM5 155561853 IC50 = 10041 nM T00407 C7FCQ9 155562154 IC50 = 79000 nM T00407 CM25ZY 155562178 IC50 = 680 nM T00407 C0JQF4 155562547 IC50 = 79.43 nM T00407 C0Y9BU 155562553 IC50 < 100 nM T00407 C2U1DO 155563442 IC50 = 709.1 nM T00407 CI3F7H 155563640 IC50 = 1584.89 nM T00407 CJ1ZK6 155563724 IC50 = 2400 nM T00407 CK0BV2 155564034 IC50 = 2511.89 nM T00407 CGWP21 155564141 IC50 = 889 nM T00407 CQK18D 155564294 IC50 = 4810000 nM T00407 C5NU8A 155564453 IC50 = 1500 nM T00407 C7ICA9 155564455 EC50 > 10000 nM T00407 CJ3ZR5 155564460 IC50 = 220 nM T00407 C47LAU 155564565 IC50 = 14.4 nM T00407 C8LF6O 155564647 IC50 = 2436 nM T00407 C7EDG4 155564694 IC50 = 10000 nM T00407 CC8O2L 155565265 IC50 = 50.12 nM T00407 C68CBM 155565352 IC50 = 25.9 nM T00407 C4VSH5 155565624 IC50 = 810.4 nM T00407 CY83NZ 155565684 Ki = 2.8 nM T00407 C17NSI 155566209 IC50 = 1960 nM T00407 CZC03T 155566251 IC50 = 176 nM T00407 CK9C6J 155566327 IC50 = 334.2 nM T00407 CXRJ70 155566441 IC50 > 50118.72 nM T00407 CJ5B1M 155566905 Ki = 2.1 nM T00407 C2PIK0 155567275 IC50 > 501187.23 nM T00407 CZK10H 155567377 IC50 > 10000 nM T00407 CM5FL1 155567534 IC50 > 50118.72 nM T00407 C8ZS0C 155567638 IC50 = 21 nM T00407 CMV75T 155567768 Ki = 1230 nM T00407 CXZG79 155567978 Ki = 1.8 nM T00407 C7C9DH 155568184 IC50 > 50118.72 nM T00407 CV9L7S 155568572 Ki = 1.3 nM T00407 CUWO65 155568681 IC50 = 68 nM T00407 C06GWZ 155568932 Ki = 24.7 nM T00407 CZ2VN0 155569163 IC50 > 50118.72 nM T00407 C48AYZ 155569378 IC50 = 800 nM T00407 CN56LR 155569534 Ki = 6.31 nM T00407 CNF0G9 155569554 IC50 = 480 nM T00407 D00DXI 135566302 Ki = 10850 nM T00407 D00XRH 91820725 IC50 = 1258.93 nM T00407 D01YSN 57345400 IC50 = 26 nM T00407 D03BTJ 15990224 IC50 = 3162.28 nM T00407 D03LIP 13953710 IC50 = 15.5 nM T00407 D03LNF 71271629 IC50 = 220 nM T00407 D03XXT 72201027 IC50 = 3200 nM T00407 D09HBR 135566899 Ki < 85 nM T00407 D09VHS 3971 IC50 = 9050 nM T00407 D09ZPM 1091852 IC50 = 79432.82 nM T00407 D0C2JS 71291068 IC50 = 92 nM T00407 D0F5TZ 91827383 IC50 = 2511.89 nM T00407 D0H3TC 54669868 IC50 = 4786.3 nM T00407 D0J3JI 90488984 IC50 = 600 nM T00407 D0J6XI 1253361 IC50 = 2500 nM T00407 D0N5BI 91668541 IC50 = 5011.87 nM T00407 D0O2RX 71624782 IC50 = 371.54 nM T00407 D0O6XT 91827373 IC50 = 3700 nM T00407 D0Q7IU 40642506 IC50 = 10400 nM T00407 D0T3WL 73010930 IC50 > 50000 nM T00407 D0T3YY 59190723 Ki = 16.7 nM T00407 D0V8MX 606801 IC50 = 4300 nM T00407 D0VC0I 5169 IC50 = 2500 nM T00407 D0WU1S 52912189 Ki = 9 nM T00407 D0Y3OO 11327430 IC50 = 1000 nM T57943 D09QDP 4380 IC50 > 100000 nM T57943 D0B7EB 36462 IC50 < 1000 nM T57943 D0S2UG 26757 IC50 > 100000 nM T57943 D01YIF 135421197 EC50 = 220 nM T57943 D04NAQ 12000240 IC50 = 6 nM T57943 D0J3SU 9847835 Ki = 1.2 nM T57943 D0U6WQ 153270 IC50 = 1300 nM T57943 D0F9FA 5311139 IC50 = 190000 nM T57943 CY0FV4 17520 IC50 = 46740 nM T57943 C13JOV 75994 EC50 > 50000 nM T57943 C6OG3J 164981 IC50 = 532.8 nM T57943 C5KHP9 200601 EC50 > 50000 nM T57943 C1BJ4H 207112 EC50 > 50000 nM T57943 CZT8Q4 263609 IC50 > 50000 nM T57943 CS15JU 337889 IC50 = 91240 nM T57943 C8MPT3 351236 IC50 = 42390 nM T57943 CJSB46 515949 IC50 = 7000 nM T57943 CD98GM 515951 IC50 > 50000 nM T57943 CAN39P 515952 IC50 = 15000 nM T57943 CNS15D 515953 IC50 = 600 nM T57943 COW5R3 608841 Ki = 4300 nM T57943 CZ52FW 611339 IC50 > 100000 nM T57943 C8ML5S 680303 IC50 = 13250 nM T57943 CAG12P 706730 IC50 = 6360 nM T57943 CI0DG1 764318 IC50 = 184700 nM T57943 C0P6TI 772300 EC50 > 10000 nM T57943 CAKL05 784811 EC50 > 10000 nM T57943 CZ5J6R 823490 EC50 > 40000 nM T57943 C4J5UE 867607 EC50 > 10000 nM T57943 CP8Y2I 870574 IC50 = 6117 nM T57943 C8D2GZ 874750 EC50 > 40000 nM T57943 CHX80I 906558 IC50 = 3 nM T57943 C9QY6A 1247468 IC50 > 50000 nM T57943 CEQ17S 1352031 IC50 = 30000 nM T57943 CJF63U 1358496 IC50 = 30000 nM T57943 CQR67C 1909002 IC50 > 100000 nM T57943 C5WKA9 2779120 IC50 = 40000 nM T57943 C64QBE 2807947 EC50 > 10000 nM T57943 CI05CP 2807954 EC50 = 790 nM T57943 C1V6CM 2821593 IC50 > 200000 nM T57943 C7CLA9 2821595 IC50 = 55000 nM T57943 C2U4HS 2821632 IC50 = 150000 nM T57943 CMP1F6 2821634 IC50 = 129000 nM T57943 CR7N4T 2821636 IC50 = 133000 nM T57943 COTB47 2821639 IC50 = 74000 nM T57943 C1JRB7 2821640 IC50 = 40000 nM T57943 C12EXP 2821660 IC50 = 82000 nM T57943 CGOH73 2821679 IC50 = 128000 nM T57943 CP1QK5 2856389 IC50 > 100000 nM T57943 C5GZ0U 2856462 IC50 > 1000000 nM T57943 CPA63I 3107941 IC50 = 29700 nM T57943 C6SO2K 3708081 IC50 > 200000 nM T57943 CF51QJ 3783248 EC50 = 440 nM T57943 C1RUH9 4246483 IC50 = 13600 nM T57943 C8RTZ6 5060109 EC50 > 50000 nM T57943 CT4YC1 5287959 IC50 = 7.95 nM T57943 C3T8NF 5288850 IC50 = 2.4 nM T57943 C0Z8HR 5288877 IC50 = 6000 nM T57943 CH9B1I 5288878 IC50 = 1735 nM T57943 CO58XD 5311161 IC50 = 43500 nM T57943 C1KR5B 5327301 Ki = 90 nM T57943 C37TKL 5327302 Ki = 200 nM T57943 C64ZMN 5327304 Ki = 50 nM T57943 C3IZ2W 5327307 Ki = 30 nM T57943 C16DTL 5327308 Ki = 120 nM T57943 C4O3QY 5327309 Ki = 20 nM T57943 C3GUM7 5327310 Ki = 40 nM T57943 CGB4W1 5327311 Ki = 480 nM T57943 C5WO0Y 5327312 Ki = 90 nM T57943 C85FLX 5327313 Ki = 70 nM T57943 CM6BP7 5327314 Ki = 160 nM T57943 CO4TA8 5327315 Ki = 60 nM T57943 CREJ96 5327316 Ki = 2500 nM T57943 C2LG6D 5327317 Ki = 380 nM T57943 CFWC38 5327318 Ki = 290 nM T57943 C56ZND 5327319 Ki = 2100 nM T57943 CI8KS4 5327320 Ki = 2400 nM T57943 CJON52 5327321 Ki = 400 nM T57943 CBF73K 5327323 Ki = 140 nM T57943 C0KGV4 5327324 Ki = 1900 nM T57943 C7TP1M 5327325 Ki = 800 nM T57943 CMV6J9 5327326 Ki = 140 nM T57943 C40MIA 5327327 Ki = 270 nM T57943 CP6KU2 5327328 Ki = 4000 nM T57943 C2A4DC 5327329 Ki = 210 nM T57943 CLN73K 5327330 Ki = 290 nM T57943 CB2F4G 5327331 Ki = 12500 nM T57943 C73USB 5327332 Ki = 4000 nM T57943 CDZH46 5327333 Ki = 20 nM T57943 C2UC8Q 5327334 Ki = 30 nM T57943 CEVM46 5327335 Ki = 240 nM T57943 CIH3Z6 5327336 Ki = 4000 nM T57943 CYSG72 5327337 Ki = 1700 nM T57943 CQU5S2 5327338 Ki = 2300 nM T57943 CMU91Y 5327339 Ki = 160 nM T57943 CAO3V1 5327340 Ki = 1700 nM T57943 C15CZY 5327341 Ki = 1900 nM T57943 CP45FJ 5327342 Ki = 1300 nM T57943 CMQ3K7 5327343 Ki = 1400 nM T57943 C3BUH9 5327344 Ki = 470 nM T57943 CET23W 5327345 Ki = 440 nM T57943 CRZ18A 5327347 Ki = 190 nM T57943 CU2N5V 5327348 Ki = 450 nM T57943 CDP82Q 5497174 IC50 = 40000 nM T57943 CR89FE 6885304 EC50 > 50000 nM T57943 C3LZX9 8027611 IC50 > 20000 nM T57943 C0LTB1 9543561 EC50 > 50000 nM T57943 CG6VT5 9543562 EC50 > 50000 nM T57943 C1GKZ4 9795048 IC50 = 18550 nM T57943 CFN2P6 9800285 Ki = 19 nM T57943 C70YBC 9800605 IC50 = 63700 nM T57943 C95HCO 9801989 IC50 = 720 nM T57943 CN24XB 9802549 IC50 = 4.6 nM T57943 CP97XI 9805997 IC50 = 2.999 nM T57943 CJ7V8I 9806866 IC50 = 130 nM T57943 CE7I9W 9806986 IC50 = 0.026 nM T57943 CYFG94 9807028 IC50 = 48 nM T57943 CD3P2F 9807170 IC50 = 0.063 nM T57943 C3S1EP 9807375 IC50 = 0.08 nM T57943 C13PRZ 9809421 IC50 = 5 nM T57943 CLTO67 9821317 IC50 = 30 nM T57943 C4XO3K 9821545 Ki = 8.3 nM T57943 CJI5T3 9823027 IC50 = 13 nM T57943 C74QTI 9823074 IC50 = 135 nM T57943 CNY5D8 9823176 IC50 = 860 nM T57943 CH4R2T 9823438 IC50 = 270 nM T57943 C1VM6Y 9823995 IC50 = 1700 nM T57943 CWI7K4 9826973 IC50 = 15000 nM T57943 CVEG78 9827110 IC50 = 400 nM T57943 C2G1HI 9827739 IC50 = 170 nM T57943 CGD27M 9834674 IC50 = 10800 nM T57943 CPUY67 9836512 EC50 = 480 nM T57943 C6S3KT 9840223 Ki = 41.8 nM T57943 CF2M1L 9840924 IC50 = 1070 nM T57943 CKMX05 9842198 IC50 = 30 nM T57943 CS50WH 9844966 IC50 = 13700 nM T57943 CA04ZU 9845902 IC50 = 320 nM T57943 C7ST4G 9848668 IC50 = 520 nM T57943 CN02PU 9849845 IC50 = 0.048 nM T57943 C5MCX4 9849846 IC50 = 0.072 nM T57943 CDC86G 9850642 IC50 = 0.16 nM T57943 CJO3A5 9851213 IC50 = 0.088 nM T57943 C56LDH 9851279 IC50 = 9 nM T57943 C6O0QH 9852052 IC50 = 0.0008 nM T57943 CO9WH2 9858488 EC50 = 830 nM T57943 CU43VF 9859323 IC50 = 10000 nM T57943 C1KJ2O 9866145 IC50 = 100 nM T57943 C6NJ3A 9866634 IC50 = 36 nM T57943 C8J1GE 9866954 IC50 = 11700 nM T57943 CD05OL 9867192 IC50 = 10 nM T57943 CMK6E5 9867709 IC50 = 1100 nM T57943 C8ZE6M 9869539 IC50 = 620 nM T57943 C5FJG7 9870833 Ki = 40 nM T57943 C2N3LE 9871540 IC50 = 0.082 nM T57943 CX17DM 9871570 IC50 = 0.018 nM T57943 CF0V7B 9871631 IC50 = 0.012 nM T57943 C3WEI5 9878404 EC50 = 760 nM T57943 C3O7PQ 9878859 EC50 = 580 nM T57943 C9C6AE 9879308 EC50 = 390 nM T57943 C3GC6F 9883721 IC50 = 18000 nM T57943 C8UI1Y 9885498 IC50 = 61 nM T57943 CJ0U5P 9885590 IC50 = 1400 nM T57943 CZM9E1 9889018 IC50 = 2500 nM T57943 C5TV0W 9889264 IC50 = 550 nM T57943 CN4V9P 9891193 IC50 = 0.37 ug.mL-1 T57943 CLQH78 9892350 IC50 = 0.071 nM T57943 CWS25H 9892517 IC50 = 270 nM T57943 CW75OE 9892652 IC50 = 0.046 nM T57943 C3YAL4 9895375 IC50 = 1.8 nM T57943 C8SRO2 9900136 IC50 = 12090 nM T57943 C8Z2BV 9900370 EC50 = 1490 nM T57943 CDB31H 9901891 EC50 = 840 nM T57943 C62LAG 9905968 IC50 = 8.8 ug.mL-1 T57943 CGC85H 9909850 IC50 = 34 nM T57943 CM4V2U 9910924 IC50 = 450 nM T57943 C8SP7V 9913141 IC50 = 5.2 nM T57943 C2DMG1 9914167 Ki = 4.8 nM T57943 CK15RJ 9916276 IC50 = 0.14 nM T57943 CNTV79 9922120 EC50 = 1450 nM T57943 C0JPU8 9922548 EC50 > 10000 nM T57943 CLNG83 9923594 EC50 = 280 nM T57943 C68DTJ 9926544 IC50 = 37 nM T57943 CA61DY 9930939 IC50 = 200 nM T57943 C0MLC1 9934739 IC50 = 4.2 nM T57943 C0D2IJ 9936767 IC50 = 0.036 nM T57943 CG90WC 9939287 IC50 = 5 nM T57943 CFCK64 9939773 IC50 = 94 nM T57943 CTB54I 9953690 IC50 = 260 nM T57943 CX6ZK9 9953736 IC50 = 36 nM T57943 C8ACO4 9955110 IC50 = 169.82 nM T57943 CN63JG 9958554 IC50 = 0.051 nM T57943 CK7ZG9 9959259 IC50 = 13400 nM T57943 C8AY0X 9965414 EC50 = 1420 nM T57943 C0G1ZI 9966013 EC50 = 290 nM T57943 C9FCA6 9967365 EC50 = 410 nM T57943 C8KS5B 9967366 EC50 = 240 nM T57943 C0HJ4M 9980296 IC50 = 390 nM T57943 C9CV0Y 10001828 IC50 = 135 nM T57943 CW4Q3N 10031194 IC50 = 73 nM T57943 CHWA42 10074552 IC50 = 130 nM T57943 CN91VE 10109081 EC50 = 1070 nM T57943 CJ3B2V 10132392 EC50 = 430 nM T57943 CI4VA9 10154401 EC50 = 1320 nM T57943 C84TLR 10155705 EC50 = 560 nM T57943 CPFJ25 10291989 EC50 = 610 nM T57943 CMR75W 10318568 IC50 = 1100 nM T57943 C0V4LP 10356503 IC50 = 4650 nM T57943 CZ3IH4 10414828 IC50 = 63 nM T57943 C8Q3KY 10459952 Ki = 70 nM T57943 CX67SZ 10826725 Ki = 130 nM T57943 CF25HL 10851609 IC50 = 909.91 nM T57943 CDX7A4 10963183 Ki = 20 nM T57943 CGZ17V 11004903 Ki = 20 nM T57943 C2GPV7 11150874 IC50 = 31.05 nM T57943 CYBT89 11179699 IC50 = 255 nM T57943 C7HSX0 11189577 IC50 = 1841 nM T57943 C6EL1S 11197291 IC50 = 31 nM T57943 CSYR59 11201705 IC50 = 23 nM T57943 CGL90K 11226974 IC50 = 27900 nM T57943 C4WU5A 11231441 IC50 = 86 nM T57943 C35RCL 11250168 IC50 = 58 nM T57943 CM8O6L 11257152 IC50 = 17 nM T57943 C0SUW1 11262077 IC50 = 5190 nM T57943 CI51QS 11282766 IC50 = 294 nM T57943 C63RSD 11307958 IC50 = 33 nM T57943 C5VCN3 11318330 IC50 = 15350 nM T57943 CH5P7O 11330337 IC50 = 352 nM T57943 C53FEL 11353611 IC50 = 362 nM T57943 CCV6T0 11374367 IC50 = 25 nM T57943 COF97S 11381357 EC50 = 380 nM T57943 C0OKW7 11381401 IC50 = 49.04 nM T57943 CAF6I3 11387099 IC50 = 1290 nM T57943 CBJ48H 11397895 IC50 = 36 nM T57943 C1WD2X 11398098 IC50 = 27 nM T57943 CK78LF 11409626 IC50 = 33 nM T57943 C2AE5Q 11442287 IC50 = 10900 nM T57943 CDK1W3 11442758 IC50 = 4 nM T57943 C4F8DC 11444079 Ki = 5.9 nM T57943 CZEJ53 11450373 EC50 = 370 nM T57943 CY96MN 11454338 IC50 = 40 nM T57943 CFW05T 11467141 IC50 = 33 nM T57943 CDT9G3 11467504 Ki = 0.0014 nM T57943 CSJ0F2 11493626 IC50 = 78 nM T57943 CQ92TS 11495091 IC50 = 3.3 nM T57943 CV4CP9 11496333 IC50 = 9.772 nM T57943 CK12ZL 11496771 IC50 = 23 nM T57943 C2O4FW 11496899 IC50 = 24.63 nM T57943 CGE2J0 11497112 IC50 = 11.22 nM T57943 CJZU36 11500289 IC50 = 176 nM T57943 CY3N0Q 11500400 IC50 = 272 nM T57943 C32ECP 11500457 IC50 = 79 nM T57943 CF7A4U 11501937 IC50 = 148 nM T57943 C6DFU0 11503023 IC50 = 191 nM T57943 C6IS9K 11509289 IC50 = 91.2 nM T57943 C6L2MY 11509300 EC50 = 1830 nM T57943 CC31QO 11509301 IC50 = 20.4 nM T57943 C70RLV 11509551 IC50 = 350 nM T57943 CS8OX7 11510566 Ki = 9 nM T57943 C7FY9B 11512139 IC50 = 12 nM T57943 C15VFG 11515586 Ki = 1.2 nM T57943 CW6PC0 11519268 IC50 = 12.3 nM T57943 CL0C9P 11525287 IC50 = 7 nM T57943 CZC5D9 11525874 IC50 = 5.754 nM T57943 CP8IY2 11529998 IC50 = 44 nM T57943 C5BNE1 11533326 IC50 = 10.3 nM T57943 CDK3Z5 11533935 Ki = 0.2 nM T57943 C3VP4D 11536658 IC50 = 262 nM T57943 CHD72T 11538521 IC50 = 66 nM T57943 C4IC7E 11541867 Ki = 0.8 nM T57943 C3USR9 11543714 IC50 = 83 nM T57943 CPFD59 11544054 IC50 = 139 nM T57943 CBC8P4 11545354 IC50 = 70 nM T57943 C3P2GZ 11548424 Ki = 1.9 nM T57943 CVX4M6 11548909 Ki = 1.2 nM T57943 CQ7US3 11552973 IC50 = 158 nM T57943 C9T4VQ 11559154 IC50 = 53 nM T57943 C6S9KI 11559640 IC50 = 201 nM T57943 CB4L2R 11560019 IC50 = 145 nM T57943 C2YN0U 11560375 IC50 = 1503 nM T57943 CPRZ67 11565014 IC50 = 164 nM T57943 C6GO1T 11566274 IC50 = 62 nM T57943 CPM0L1 11567908 IC50 = 14.83 nM T57943 CURG08 11572178 IC50 = 191 nM T57943 CDU5C8 11572524 IC50 = 92 nM T57943 C17OJS 11572844 IC50 = 68 nM T57943 CNUG62 11574810 IC50 = 104 nM T57943 C8RNL1 11576032 IC50 = 15 nM T57943 CM96SG 11576187 IC50 = 59 nM T57943 CF0V3P 11576540 IC50 = 5.2 nM T57943 C1T9DY 11576622 IC50 = 29.2 nM T57943 C03KPR 11576852 IC50 = 12.1 nM T57943 C72DIR 11577083 IC50 = 81 nM T57943 C89CAJ 11581298 IC50 = 210 nM T57943 CN67DR 11583840 IC50 = 8.71 nM T57943 CPD0M8 11584106 IC50 = 21.3 nM T57943 CM8PD5 11588119 IC50 = 124 nM T57943 C70WFH 11590421 IC50 = 4.99 nM T57943 CP0BO4 11591156 IC50 = 13.83 nM T57943 CL16IM 11591540 IC50 = 3.9 nM T57943 CE2TX6 11591919 Ki = 8 nM T57943 CLDJ71 11594984 IC50 = 437 nM T57943 CTIC48 11597226 IC50 = 16 nM T57943 CG4Z9A 11598106 IC50 = 8.3 nM T57943 CI20RN 11604867 IC50 = 2524 nM T57943 CEU02V 11609502 IC50 = 103 nM T57943 C9OZ5P 11611743 IC50 = 13.61 nM T57943 CV6MF1 11614728 Ki > 5000 nM T57943 C40XHV 11615842 IC50 = 193 nM T57943 CK81HR 11619252 IC50 = 37 nM T57943 CFP19E 11619968 IC50 = 10.9 nM T57943 C03KFC 11623986 IC50 = 763 nM T57943 C5SP7Y 11624054 IC50 = 384 nM T57943 CT7ZF5 11624098 IC50 = 59 nM T57943 CA5BX8 11624232 IC50 = 54 nM T57943 CA0LH6 11624920 IC50 = 286.7 nM T57943 CJV73T 11626641 IC50 = 7.81 nM T57943 C0UG4X 11626852 IC50 = 1.29 nM T57943 CK7WY3 11626961 IC50 = 10.77 nM T57943 CEY39D 11628992 Ki = 8.6 nM T57943 C6UAV3 11632008 IC50 = 40 nM T57943 C6Y5MG 11634372 IC50 = 9.333 nM T57943 CM2U8T 11634523 IC50 = 37 nM T57943 CKJE92 11634649 IC50 = 9.1 nM T57943 C4QB6F 11635889 IC50 > 10000 nM T57943 CG2C6A 11638464 IC50 = 150 nM T57943 C91JNO 11639020 IC50 = 25 nM T57943 CREY96 11639401 IC50 = 44 nM T57943 C7Z0YL 11640020 IC50 = 1338 nM T57943 C4MCW2 11646889 IC50 = 113 nM T57943 C2KFU3 11647018 IC50 = 23.44 nM T57943 CM59UT 11649267 IC50 = 14.32 nM T57943 CS0MQ7 11652262 IC50 = 110 nM T57943 C17AMN 11652763 IC50 = 199 nM T57943 CH20JE 11652994 IC50 = 1380 nM T57943 CL74QK 11654098 IC50 = 148 nM T57943 CW5R3S 11661117 IC50 = 6 nM T57943 CN32TX 11664423 Ki = 9.8 nM T57943 C4UH0Z 11670824 IC50 = 82 nM T57943 CUD05C 11670894 IC50 = 4.365 nM T57943 C26RQJ 11681876 IC50 = 356 nM T57943 CX43CE 11682171 IC50 = 364 nM T57943 C5X0KG 11682504 IC50 = 2394 nM T57943 C5D3KH 11683258 IC50 = 71 nM T57943 CR4OK8 11684562 IC50 = 4.43 nM T57943 CX97NT 11684618 IC50 = 8.318 nM T57943 CY18SQ 11695300 IC50 = 99 nM T57943 CI23AO 11695775 IC50 = 118 nM T57943 CBO30C 11698907 IC50 = 30 nM T57943 CBS3M1 11699168 IC50 = 10.14 nM T57943 C05YRV 11699954 Ki = 12.6 nM T57943 CKEX64 11700402 Ki = 12.6 nM T57943 C48UXS 11702074 IC50 = 140 nM T57943 CK08NC 11702560 IC50 = 96 nM T57943 CQ42JX 11705447 IC50 = 7.18 nM T57943 C89COT 11705942 IC50 = 8.318 nM T57943 C16WIO 11711242 IC50 = 55 nM T57943 C29UWG 11712170 IC50 = 2.4 nM T57943 C86PAH 11712912 Ki = 4 nM T57943 CY90EM 11712953 IC50 > 10000 nM T57943 CNV75J 11713799 IC50 > 10000 nM T57943 CY1LN0 11719933 IC50 = 2.32 nM T57943 C7QK5F 11755713 IC50 = 310 nM T57943 CTY2B0 12223544 IC50 = 22720 nM T57943 CLV92M 12390050 IC50 > 45000 nM T57943 CY56QF 13369486 Ki = 732120 nM T57943 C4P5HI 14490061 Ki > 1000000 nM T57943 CRWS56 16046172 IC50 > 10000 nM T57943 C8XJB3 16098559 Ki = 1400 nM T57943 CT2WL8 16098564 Ki = 1000 nM T57943 CN9JO5 16098566 Ki = 1100 nM T57943 C7YI1R 16725993 IC50 = 19390 nM T57943 CXH9M5 16749067 IC50 = 272 nM T57943 C2DJ5W 16749068 IC50 = 3.89 nM T57943 COM07G 16749069 IC50 = 119.3 nM T57943 CPG8Q0 16749161 IC50 = 31.8 nM T57943 CG84TK 16749162 IC50 = 7.6 nM T57943 CT3HD1 16749163 IC50 = 7.8 nM T57943 CZM4X2 16749164 IC50 = 7.8 nM T57943 CUZ8N4 16749267 IC50 = 9.85 nM T57943 CMEK96 16749268 IC50 = 3.6 nM T57943 C01HBN 16749269 IC50 = 27.8 nM T57943 CWG3C8 16749270 IC50 = 20.1 nM T57943 C8R3GD 16749271 IC50 = 5.1 nM T57943 CDT59W 22422581 IC50 = 8110 nM T57943 C6YI1C 22456688 IC50 = 140000 nM T57943 C0MSR3 22456709 IC50 = 69.98 nM T57943 CRW91K 22456716 IC50 = 31 nM T57943 CB35YF 22456736 IC50 = 169.82 nM T57943 CH6S9A 23460501 IC50 = 1580 nM T57943 CX61VS 23645111 Ki = 6400 nM T57943 CEQT03 23645112 Ki = 1800 nM T57943 C7TBJ2 23645113 Ki = 800 nM T57943 C68GZW 23645114 Ki = 700 nM T57943 CNBG96 23645115 Ki = 600 nM T57943 C6GPY5 23645116 Ki = 4400 nM T57943 C2R0TP 23645117 Ki = 1300 nM T57943 C8R6IY 23645118 Ki = 100 nM T57943 CU2R0S 23645119 Ki = 200 nM T57943 CSTU86 23645120 Ki = 200 nM T57943 CZM4X5 23645121 Ki = 200 nM T57943 CVP6Q9 23645122 Ki = 200 nM T57943 CDB87T 23645123 Ki = 200 nM T57943 CX7MK2 23645124 Ki = 100 nM T57943 CE8S9M 23645125 Ki = 600 nM T57943 CY5KJ2 23645126 Ki = 70 nM T57943 CV4S9U 23645127 Ki = 100 nM T57943 C5S4TM 23645128 Ki = 5800 nM T57943 CCA03Z 23645129 Ki = 2000 nM T57943 C38PNH 23645130 Ki = 6800 nM T57943 CEA91D 23645131 Ki = 1400 nM T57943 C06OPL 23645134 Ki = 1800 nM T57943 C07DJM 23645135 Ki = 400 nM T57943 C6KT2X 23645136 Ki = 600 nM T57943 COL58N 23645137 Ki = 300 nM T57943 C23BAX 23645138 Ki = 3300 nM T57943 CXP1U0 23645139 Ki = 1000 nM T57943 C81OBV 23645140 Ki = 4000 nM T57943 C5S0CL 23645141 Ki = 300 nM T57943 CK9ND4 23645142 Ki = 300 nM T57943 CE4D1P 23645146 IC50 = 62800 nM T57943 CGM6N3 23645147 IC50 = 37100 nM T57943 C4BOD6 23645148 IC50 = 2500 nM T57943 CHWV78 23645149 IC50 = 460 nM T57943 CBOS13 23645150 IC50 = 23300 nM T57943 C8FYT2 23645151 IC50 = 5500 nM T57943 CZA29P 23645152 IC50 = 1080 nM T57943 CZUM37 23645153 IC50 = 2540 nM T57943 C3KBV7 23645155 IC50 = 90 nM T57943 C10ZXB 23645156 IC50 = 360 nM T57943 C08SKU 23645158 IC50 = 16 nM T57943 CZ1BW9 23645159 IC50 = 33 nM T57943 C9BNV1 23645160 IC50 = 200 nM T57943 C1HWV6 23645161 IC50 = 21 nM T57943 C81XEB 23645162 IC50 = 23 nM T57943 CW9HL5 23645230 IC50 = 60 nM T57943 C5G2IL 23645238 IC50 = 341 nM T57943 C74OPE 23645239 IC50 = 746 nM T57943 CK7B2A 23645240 IC50 = 41 nM T57943 C8YA0T 23645241 IC50 = 100 nM T57943 C8J7UY 23645242 IC50 = 330 nM T57943 C3MGC1 23645243 IC50 = 118 nM T57943 CLSU45 23645244 IC50 = 425 nM T57943 C95KHP 23645245 IC50 = 85 nM T57943 C08UYG 23645246 IC50 = 1295 nM T57943 C6YEO7 23645247 IC50 = 2020 nM T57943 CFH23D 23645248 IC50 = 467 nM T57943 CY0M3Z 23645249 IC50 = 160 nM T57943 C4TIM0 23645250 IC50 = 146 nM T57943 CZ9HT6 23645253 IC50 = 10 nM T57943 C1CB4I 23645256 IC50 = 23000 nM T57943 CZIW07 23645257 IC50 = 55000 nM T57943 C4L0GF 23645258 IC50 > 200000 nM T57943 CPN0E7 23645259 IC50 = 96900 nM T57943 CV3GC2 23645260 IC50 = 1200 nM T57943 C9XVN2 23645261 IC50 = 410 nM T57943 CC7ZF1 23645262 IC50 = 250 nM T57943 CRA3C1 23645263 IC50 = 130 nM T57943 CXPF97 23645264 IC50 = 300 nM T57943 C4PN3E 23645265 IC50 = 170 nM T57943 CQAN78 23645266 IC50 = 340 nM T57943 C68KUV 23645305 IC50 = 9.17 nM T57943 CZ59CM 23645306 IC50 = 140 nM T57943 CNU1R6 23645307 IC50 = 83 nM T57943 C8WF2G 23645308 IC50 = 210 nM T57943 CBSA54 23645309 IC50 = 53 nM T57943 CL1CX8 23672868 IC50 = 140 nM T57943 C7IQO2 24901498 IC50 = 15 nM T57943 CTI80F 25178948 EC50 = 17 nM T57943 C2GI4J 25178949 EC50 = 16.8 nM T57943 CQ2GM9 25178950 EC50 = 2.3 nM T57943 C4GFV6 25179140 EC50 = 50.1 nM T57943 CYL36B 25179141 EC50 = 0.5 nM T57943 CGC69Q 25179143 EC50 = 199.5 nM T57943 C27YJF 25179144 EC50 = 16.7 nM T57943 C2YTB7 25179145 EC50 = 12.6 nM T57943 C6GTV3 25179324 EC50 = 26.1 nM T57943 CIC46T 25179513 EC50 = 12.4 nM T57943 CK96WB 25179514 EC50 = 5.5 nM T57943 CGX78D 25217029 IC50 = 6 nM T57943 CW2L9Q 25217030 IC50 = 7.5 nM T57943 C8UTC4 25217031 IC50 = 7.1 nM T57943 CZ43KQ 25217032 IC50 = 18.3 nM T57943 C2P9NI 25217145 EC50 = 2000 nM T57943 C8C9XU 42618276 IC50 = 1430 nM T57943 CFO93N 42618277 IC50 = 1023.29 nM T57943 CS1KQ0 42618278 IC50 = 583 nM T57943 CVI16X 42618279 IC50 = 1405 nM T57943 C3MRA0 42618280 IC50 = 529 nM T57943 C8UO9S 42618281 IC50 = 4700 nM T57943 C68NPR 42618282 IC50 = 4633 nM T57943 CL41SD 42618283 IC50 = 1550 nM T57943 CJ7U2E 42618284 IC50 = 1454 nM T57943 CZL8C7 42618285 IC50 = 1672 nM T57943 CNIQ28 42618286 IC50 = 1993 nM T57943 C91OMB 42618287 IC50 = 114 nM T57943 C5AC1L 42618288 IC50 = 323 nM T57943 CFU5T2 42618289 IC50 = 718 nM T57943 CK9H3M 42618290 IC50 = 365 nM T57943 CV4H2J 42618291 IC50 = 671 nM T57943 C7VPU3 42618292 IC50 = 673 nM T57943 C6R2FM 42618293 IC50 = 724 nM T57943 C0YOE3 43816622 IC50 = 34000 nM T57943 C4QOV7 44157030 IC50 = 5.3 nM T57943 CGB3E4 44157031 IC50 = 29 nM T57943 CT2B8Z 44157032 IC50 = 25 nM T57943 CT7VO2 44157085 IC50 = 151 nM T57943 CWMU91 44157086 IC50 = 3.6 nM T57943 C6LZ5Y 44157087 IC50 = 23 nM T57943 CYSJ79 44157089 IC50 = 6.6 nM T57943 CMX7W1 44157090 IC50 = 42 nM T57943 C35DAU 44158016 IC50 = 1880 nM T57943 C7B3VE 44158086 IC50 = 43 nM T57943 C20WEJ 44158089 IC50 = 19 nM T57943 C68KOD 44158154 IC50 = 80 nM T57943 C4C1RU 44158155 IC50 = 145 nM T57943 CN1YR9 44158157 IC50 = 11 nM T57943 C80XPD 44158237 IC50 = 275 nM T57943 CN09UV 44158238 IC50 = 25 nM T57943 CT9DF4 44158240 IC50 = 31 nM T57943 CHDF62 44158242 IC50 = 74 nM T57943 CS6X1C 44158325 IC50 = 9.3 nM T57943 C17TEZ 44158326 IC50 = 10 nM T57943 CZ0VT3 44158328 IC50 = 17 nM T57943 C4NLH9 44204064 IC50 = 19140 nM T57943 CRN06H 44204163 IC50 = 28180 nM T57943 C2G0OC 44204165 IC50 = 26800 nM T57943 C0GA8R 44204268 IC50 = 32320 nM T57943 C6T8PR 44204269 IC50 = 11330 nM T57943 C6TOU8 44204270 IC50 > 45000 nM T57943 CC31OK 44204271 IC50 = 16580 nM T57943 C8AP6D 44204365 IC50 = 27660 nM T57943 CZ80VE 44204459 IC50 = 19670 nM T57943 CHXU65 44204460 IC50 = 40960 nM T57943 C5DGZ4 44283428 IC50 = 438 nM T57943 CV6KT8 44303728 IC50 = 410 nM T57943 CHZ78B 44303973 IC50 = 44 nM T57943 CD8WB9 44304162 IC50 = 5495.41 nM T57943 CV7O8U 44309729 Ki = 202 nM T57943 C9RLK1 44309811 Ki = 71 nM T57943 C2VW1E 44309957 Ki = 143 nM T57943 CP38YD 44325861 IC50 > 100000 nM T57943 CK89PV 44325864 IC50 > 10000 nM T57943 C0CB5F 44325871 IC50 > 100000 nM T57943 CR0D8P 44325874 IC50 > 10000 nM T57943 CM10IP 44325901 IC50 = 47000 nM T57943 CE6IX1 44325902 IC50 > 10000 nM T57943 CU36WF 44325934 IC50 = 18 nM T57943 CR46LI 44325936 IC50 = 86000 nM T57943 C8J6DK 44325943 IC50 > 10000 nM T57943 CG42XT 44325947 IC50 = 3490 nM T57943 C67TMU 44325972 IC50 = 14000 nM T57943 C93VXY 44325973 IC50 = 53000 nM T57943 CAB39E 44331552 IC50 = 375 nM T57943 CE0FW4 44331565 IC50 = 357 nM T57943 C8SZN9 44331566 IC50 = 231 nM T57943 CMFW61 44331567 IC50 = 263 nM T57943 CHYL38 44331577 IC50 = 837 nM T57943 C1I9QH 44331578 IC50 = 346 nM T57943 C4VGZ1 44331579 IC50 = 490 nM T57943 CRZ01H 44331580 IC50 = 763 nM T57943 CFOR90 44331674 IC50 = 311 nM T57943 CK7VI8 44331675 IC50 = 95 nM T57943 CH7GS4 44331676 IC50 = 3400 nM T57943 C4FOD3 44331693 IC50 = 419 nM T57943 CJY5L2 44331739 IC50 = 162 nM T57943 C8N2GQ 44331740 IC50 = 324 nM T57943 CW9K4Q 44331815 IC50 = 197 nM T57943 CT76DG 44331816 IC50 = 570 nM T57943 CC70GF 44331830 IC50 = 137 nM T57943 CNJ19L 44331876 IC50 = 849 nM T57943 C46IPA 44331879 IC50 = 6740 nM T57943 CP0Y8M 44331898 IC50 = 1.2 nM T57943 CF3R6W 44331908 IC50 = 5060 nM T57943 C0S8LV 44331910 IC50 = 2.3 nM T57943 CTM5W1 44331914 IC50 = 3.8 nM T57943 C0YZ9O 44331915 IC50 = 21 nM T57943 CPZ7Q2 44331933 IC50 = 853 nM T57943 C4NK1S 44331942 IC50 = 3.5 nM T57943 CXKY19 44331943 IC50 = 940 nM T57943 C3FC8D 44331944 IC50 > 10000 nM T57943 CH1ZF2 44331953 IC50 = 320 nM T57943 C0QJ8V 44331957 IC50 = 4400 nM T57943 C1HBX6 44331963 IC50 = 3470 nM T57943 C7UXK5 44331964 IC50 = 1750 nM T57943 C42PGN 44331965 IC50 = 230 nM T57943 C5J7KX 44331966 IC50 = 3400 nM T57943 CG83FS 44331967 IC50 = 147 nM T57943 CGAJ95 44331977 IC50 = 401 nM T57943 CCYX84 44331980 IC50 = 355 nM T57943 C5UIO2 44331987 IC50 = 528 nM T57943 C0PM5C 44332004 IC50 = 1590 nM T57943 C4ENB1 44332005 IC50 = 207 nM T57943 CFK4Z1 44332024 IC50 = 376 nM T57943 CTM3G2 44332026 IC50 = 412 nM T57943 C48ZEW 44332028 IC50 = 232 nM T57943 C30MKG 44332029 IC50 = 1570 nM T57943 C7OS9X 44332050 IC50 = 222 nM T57943 C9Y6NP 44332051 IC50 = 1390 nM T57943 C0VGF8 44332058 IC50 = 474 nM T57943 CQU84D 44332068 IC50 = 545 nM T57943 CBL91D 44332078 IC50 = 319 nM T57943 C4VCM3 44332093 IC50 = 910 nM T57943 C92QVT 44332108 IC50 = 195 nM T57943 CQLZ09 44332109 IC50 = 4810 nM T57943 C4CUL6 44332112 IC50 = 1920 nM T57943 CN2YM6 44332113 IC50 = 731 nM T57943 C4CY8K 44332118 IC50 = 1550 nM T57943 CXZ2N1 44332120 IC50 = 407 nM T57943 CD56PK 44332121 IC50 = 412 nM T57943 C5A6OJ 44332128 IC50 = 2760 nM T57943 C6IZ2R 44332129 IC50 = 269 nM T57943 C5DY0G 44332136 IC50 = 54 nM T57943 CQ1K9H 44332311 IC50 = 13 nM T57943 C9LOS2 44332330 IC50 = 59 nM T57943 C2U6GB 44332331 IC50 = 1420 nM T57943 CH01QW 44332332 IC50 = 967 nM T57943 CL92AF 44343519 Ki = 2800 nM T57943 C8OH2L 44343577 Ki = 20 nM T57943 C7CKS0 44343614 Ki ~ 50000 nM T57943 C9H1OB 44346275 Ki = 100 nM T57943 CH47FA 44346459 Ki = 7.1 nM T57943 C6W2BJ 44346460 Ki = 90 nM T57943 CBU4P3 44364553 Ki = 410 nM T57943 C8D5TB 44364680 Ki = 30 nM T57943 CV23MO 44389236 IC50 = 0.11 nM T57943 C2I3VJ 44389240 IC50 = 0.0003 nM T57943 CI89LR 44389245 IC50 = 0.042 nM T57943 CR7VM8 44389295 IC50 = 0.31 nM T57943 CU5VW3 44389297 IC50 = 0.014 nM T57943 C5P8TU 44389299 IC50 = 0.1 nM T57943 C5YC0O 44389306 IC50 = 0.033 nM T57943 C1FMX8 44389307 IC50 = 0.12 nM T57943 CB6US3 44389310 IC50 = 0.053 nM T57943 CC8S0I 44389315 IC50 = 0.0079 nM T57943 CEO19T 44389316 IC50 = 0.026 nM T57943 CRC82Z 44389318 IC50 = 0.19 nM T57943 CPE0S2 44389319 IC50 = 0.021 nM T57943 CC8MG3 44389324 IC50 = 0.005 nM T57943 C9X1RJ 44389325 IC50 = 0.078 nM T57943 CF0CN3 44389326 IC50 = 0.017 nM T57943 C7LQP0 44389331 IC50 = 0.023 nM T57943 CEQ2L1 44389335 IC50 = 0.14 nM T57943 C9C3JB 44389337 IC50 = 0.015 nM T57943 CU0I3N 44389338 IC50 = 0.013 nM T57943 CALT41 44389340 IC50 = 0.064 nM T57943 C5LO3T 44389347 IC50 = 0.014 nM T57943 CJA5K7 44389348 IC50 = 0.056 nM T57943 C2WS9G 44389351 IC50 = 0.014 nM T57943 CEH8Z5 44389369 IC50 = 0.011 nM T57943 CBJ15U 44389458 IC50 = 0.013 nM T57943 C2OU7Z 44389483 IC50 = 0.009 nM T57943 CA81WI 44389513 IC50 = 0.006 nM T57943 CL4G2Y 44389531 IC50 = 0.013 nM T57943 CX5Y3A 44389532 IC50 = 0.006 nM T57943 CEH02Q 44389544 IC50 = 0.016 nM T57943 CXN03I 44389545 IC50 = 0.0001 nM T57943 C1B7RY 44389673 IC50 = 70 nM T57943 CVA5B9 44389696 IC50 = 5 nM T57943 C6TP5D 44389700 IC50 = 12 nM T57943 C14QSK 44389749 IC50 = 20 nM T57943 CEIG09 44389792 IC50 = 50 nM T57943 CS7CK6 44389810 IC50 = 70 nM T57943 CYX73C 44389811 IC50 = 20 nM T57943 CXI7P8 44389828 IC50 = 6 nM T57943 C1E3DM 44389837 IC50 = 19 nM T57943 CHF54P 44389850 IC50 = 14 nM T57943 C8XMU0 44389851 IC50 = 14 nM T57943 CL79GW 44389871 IC50 = 66 nM T57943 CQPY50 44391346 IC50 = 80 nM T57943 CJQE23 44391364 IC50 = 176 nM T57943 CE3YN5 44391369 IC50 = 9445 nM T57943 CWVF04 44391384 IC50 = 274 nM T57943 C0J6SU 44391388 IC50 = 181 nM T57943 C24KOF 44391455 IC50 = 323 nM T57943 CD02TW 44391469 IC50 = 55 nM T57943 CA58XR 44391530 IC50 = 29 nM T57943 CU3ZB5 44391569 IC50 = 5 nM T57943 CI7F3G 44391602 IC50 = 16 nM T57943 CL73OE 44391603 IC50 = 12 nM T57943 CIU0P1 44391632 IC50 = 16 nM T57943 CXP61L 44395180 IC50 = 30 nM T57943 C3IUN4 44395181 IC50 = 110 nM T57943 CK28DO 44395208 IC50 = 98 nM T57943 CVH70D 44395211 IC50 = 35 nM T57943 C6YXO7 44395264 IC50 = 35 nM T57943 C0AVD6 44395270 IC50 = 30 nM T57943 C8KPD4 44395272 IC50 = 38 nM T57943 CCAM51 44395277 IC50 = 29 nM T57943 C65ISH 44395301 IC50 = 21 nM T57943 C5NP8T 44395302 IC50 = 15 nM T57943 CX6A5C 44395318 IC50 = 46 nM T57943 CY39WN 44395320 IC50 = 28 nM T57943 C2OW3J 44395397 IC50 = 33 nM T57943 CJ75BC 44395398 IC50 = 50 nM T57943 C8AHU6 44395469 IC50 = 250 nM T57943 CVN12E 44395477 IC50 = 81 nM T57943 C4K8RM 44398851 EC50 = 1970 nM T57943 C9VQ1J 44398919 EC50 > 10000 nM T57943 C5J4LV 44403257 IC50 > 10000 nM T57943 CYNX83 44403316 IC50 > 10000 nM T57943 CAGR97 44403319 IC50 > 10000 nM T57943 CWQ21I 44403320 IC50 > 10000 nM T57943 C5P9KT 44403321 IC50 > 10000 nM T57943 CB2E3T 44403325 IC50 > 10000 nM T57943 CAU6G0 44404870 IC50 = 4394 nM T57943 CU4N7M 44404871 IC50 = 10000 nM T57943 C3RL0N 44404877 IC50 = 2293 nM T57943 CGQ1U4 44404931 IC50 = 10000 nM T57943 CKU1S0 44404937 IC50 = 10000 nM T57943 CO38AJ 44405528 IC50 > 10000 nM T57943 CBY58A 44405529 IC50 > 10000 nM T57943 CVJ8Z3 44405532 IC50 > 10000 nM T57943 CHG69W 44405540 IC50 > 10000 nM T57943 CZ8Y2S 44405566 IC50 > 10000 nM T57943 C6X1JT 44405629 IC50 = 3260 nM T57943 CK62FC 44405634 IC50 > 10000 nM T57943 COXU97 44405637 IC50 > 10000 nM T57943 CGV2B4 44405663 IC50 > 10000 nM T57943 CFX81S 44405672 IC50 = 8070 nM T57943 CS40LN 44405689 IC50 > 10000 nM T57943 C2MOF9 44405695 IC50 = 4850 nM T57943 CYG86L 44405707 IC50 > 10000 nM T57943 CMUS37 44405733 IC50 > 10000 nM T57943 CJ07FL 44405737 IC50 > 10000 nM T57943 C1VY3T 44405740 IC50 > 10000 nM T57943 C0DL8M 44405752 IC50 > 10000 nM T57943 CB7V6W 44405784 IC50 > 10000 nM T57943 C1VW8E 44405799 IC50 > 10000 nM T57943 CH6CN5 44405800 IC50 > 10000 nM T57943 C8EK9W 44405805 IC50 > 10000 nM T57943 CWP51F 44405816 IC50 > 10000 nM T57943 CEY48X 44405818 IC50 > 10000 nM T57943 CXA87L 44405820 IC50 > 10000 nM T57943 CM2GJ1 44405827 IC50 > 10000 nM T57943 CAY57C 44405829 IC50 > 10000 nM T57943 C7LEI3 44405837 IC50 > 10000 nM T57943 CUY3M1 44414212 IC50 > 10000 nM T57943 C79OFE 44414311 IC50 > 10000 nM T57943 CFL7O1 44414418 IC50 > 10000 nM T57943 C2DIQ3 44414439 IC50 > 10000 nM T57943 C9Q4KR 44414440 IC50 > 10000 nM T57943 C0FQ1E 44414442 IC50 > 10000 nM T57943 C50NAG 44414456 IC50 > 10000 nM T57943 C34DMY 44414457 IC50 > 10000 nM T57943 CV0EW7 44414458 IC50 > 10000 nM T57943 CL29BC 44414459 IC50 > 10000 nM T57943 CV96AO 44414484 IC50 > 10000 nM T57943 C9P7ZA 44414485 IC50 > 10000 nM T57943 C4GWP5 44414501 IC50 > 10000 nM T57943 CY0VU1 44414502 IC50 > 10000 nM T57943 C8H5YL 44414541 IC50 > 10000 nM T57943 CW45EL 44414543 IC50 > 10000 nM T57943 CB0M5Q 44414572 IC50 > 10000 nM T57943 CXEH76 44414573 IC50 > 10000 nM T57943 CMI4Z9 44414574 IC50 > 10000 nM T57943 CJT30G 44414592 IC50 > 10000 nM T57943 CIQ36K 44414642 IC50 > 10000 nM T57943 CW0MH5 44416221 IC50 > 10000 nM T57943 COS6D2 44416249 IC50 > 10000 nM T57943 CL6YM3 44416250 IC50 > 10000 nM T57943 CL8IC5 44416262 IC50 > 10000 nM T57943 C21FST 44416320 IC50 > 10000 nM T57943 C3FO6V 44416321 IC50 > 10000 nM T57943 CN91HB 44416330 IC50 > 10000 nM T57943 CF6J2T 44416331 IC50 > 10000 nM T57943 CJ6QG4 44417479 Ki = 23.5 nM T57943 CTH8Y6 44418959 Ki = 1500 nM T57943 C7RX9I 44418960 Ki = 840 nM T57943 C36TBW 44421354 Ki = 3.2 nM T57943 C0YBP2 44428506 IC50 > 10000 nM T57943 CY3K9C 44428508 IC50 > 10000 nM T57943 CF2NM3 44428511 IC50 > 10000 nM T57943 CD9VU2 44428513 IC50 > 10000 nM T57943 CT8R6X 44428515 IC50 > 10000 nM T57943 CS87UF 44428517 IC50 > 10000 nM T57943 C12AHI 44428519 IC50 > 10000 nM T57943 CWG6S2 44428521 IC50 > 10000 nM T57943 CYHS50 44428523 IC50 = 7510 nM T57943 CERS10 44428524 IC50 > 10000 nM T57943 C2Q0FD 44428525 IC50 > 10000 nM T57943 C9R5MT 44428526 IC50 > 10000 nM T57943 C3CY9O 44428527 IC50 > 10000 nM T57943 CM50ES 44428528 IC50 > 10000 nM T57943 CP3XJ0 44428530 IC50 = 6810 nM T57943 C62JNP 44428532 IC50 = 1698 nM T57943 C5AE0W 44428534 IC50 = 3372 nM T57943 CE0V2J 44428536 IC50 = 1079 nM T57943 CL6K0W 44428539 IC50 = 1128 nM T57943 CFOM71 44434242 IC50 = 250 nM T57943 CU5V6D 44434244 IC50 = 1900 nM T57943 C1IAN0 44434245 IC50 = 210 nM T57943 CEK2Q4 44434246 IC50 = 100 nM T57943 C79AWI 44434247 IC50 = 410 nM T57943 CRD38M 44434248 IC50 = 340 nM T57943 CXR1V5 44434249 IC50 = 33 nM T57943 C31JIN 44438441 IC50 = 100 nM T57943 CKI30F 44438442 IC50 = 50 nM T57943 CNO1C0 44438443 IC50 = 160 nM T57943 CI1G7O 44438444 IC50 = 28 nM T57943 COP9N6 44458872 IC50 = 14000 nM T57943 C2BFJ9 44458873 IC50 = 600 nM T57943 CILG21 44458884 IC50 = 1600 nM T57943 C74XDG 44458904 IC50 = 150 nM T57943 CSN16L 44458905 IC50 = 100 nM T57943 CSYP46 44458906 IC50 = 100 nM T57943 C7FQT6 44458923 IC50 = 100 nM T57943 CMK19V 44458936 IC50 = 400 nM T57943 C4DXH1 44458937 IC50 = 1900 nM T57943 C7PTF4 44458938 IC50 = 2300 nM T57943 CJ8B0M 44458978 IC50 = 200 nM T57943 C9SC0Y 44461387 IC50 = 3 nM T57943 C9SN7W 44572193 IC50 > 100000 nM T57943 C17DXL 44572194 IC50 > 100000 nM T57943 CMJN04 44572195 IC50 = 13.3 nM T57943 CV69UW 44572196 IC50 = 359 nM T57943 C2MY8P 44572210 IC50 = 213 nM T57943 CUD5Q6 44572270 IC50 = 66 nM T57943 C4K3YQ 44572673 IC50 = 183 nM T57943 C3LYN7 44572674 IC50 = 90 nM T57943 CK4P3D 44572710 IC50 = 78 nM T57943 C62IOT 44572711 IC50 = 230 nM T57943 CZMC41 44572712 IC50 = 187 nM T57943 CZ6Y1F 44572713 IC50 = 30 nM T57943 CL5E3R 44572714 IC50 = 56 nM T57943 C1TD7H 44572774 IC50 = 1840 nM T57943 CJQ0M7 44572775 IC50 = 5120 nM T57943 CRY8Z1 44572776 IC50 = 41 nM T57943 C9YZ1J 44572777 IC50 = 499 nM T57943 C4PZ2Q 44572967 IC50 = 83 nM T57943 CH6N1M 44572968 IC50 = 191 nM T57943 CI71AG 44572969 IC50 = 82 nM T57943 CNR7O3 44572970 IC50 = 43 nM T57943 C1IZ3B 44573088 IC50 > 100000 nM T57943 CRK8D6 44573089 IC50 = 6080 nM T57943 CA4TE6 44573090 IC50 = 60900 nM T57943 CA7QH2 44573091 IC50 = 9430 nM T57943 C9QKG7 45105112 IC50 = 76 nM T57943 C3DRB6 45496892 IC50 > 200000 nM T57943 CV2I9L 46226751 IC50 = 43.63 nM T57943 C49VCB 46226760 IC50 = 10.24 nM T57943 CBJ7L2 46226763 IC50 = 12.57 nM T57943 C3Z5CV 46830074 IC50 > 200000 nM T57943 CPK5F2 46933019 IC50 = 453000 nM T57943 C4KTH5 46933020 IC50 = 434600 nM T57943 CV34ZB 46933021 IC50 = 16200 nM T57943 C3HRL2 46933163 IC50 = 23700 nM T57943 CUR1F7 46933318 IC50 = 343000 nM T57943 CON93T 46933459 IC50 = 387900 nM T57943 CL4I1F 46933460 IC50 = 185400 nM T57943 CM5T3U 46933463 IC50 = 30500 nM T57943 C7JW2B 46933464 IC50 = 69100 nM T57943 C82LPS 46933615 IC50 = 28800 nM T57943 CDY2W5 49796910 Ki = 0.005 nM T57943 CVR4C5 49796927 IC50 = 100 nM T57943 C0HMT1 49797331 IC50 = 6.6 nM T57943 C5A0BY 51346911 IC50 = 9 nM T57943 CWD7M3 51346912 Ki = 14.5 nM T57943 CN8L7W 51723030 IC50 = 50000 nM T57943 C3M2BW 52918163 EC50 = 380 nM T57943 CF24IM 52918177 EC50 = 390 nM T57943 CR9I7F 52918178 EC50 = 350 nM T57943 C2VPU1 52918179 EC50 = 420 nM T57943 CZF7K4 52943262 IC50 = 655800 nM T57943 C47TKY 52948065 IC50 = 35300 nM T57943 CO2LY5 53317588 IC50 = 44 nM T57943 C0VFY3 53320385 IC50 = 21 nM T57943 C6IK7A 53321501 IC50 = 243 nM T57943 CP31HE 53321502 IC50 = 136 nM T57943 CM30AE 53322828 IC50 = 18 nM T57943 C4EI5K 53322829 IC50 = 30 nM T57943 CB6OC8 53322830 IC50 = 267 nM T57943 C0YUM8 53324162 IC50 = 21 nM T57943 CXO2W5 53324185 IC50 = 207 nM T57943 C9QAG4 53325459 IC50 = 70 nM T57943 C7VX5Z 53325522 IC50 = 136 nM T57943 CFR32D 53326718 IC50 = 23 nM T57943 CB1U5D 53326719 IC50 = 103 nM T57943 C1W6GK 53326720 IC50 = 213 nM T57943 C8Z2TQ 54580470 EC50 = 2150 nM T57943 CMU0B4 54581481 EC50 = 1690 nM T57943 CCS8Y3 54581987 IC50 = 23.3 nM T57943 CJEP38 54582484 EC50 = 1300 nM T57943 C61NWL 54582924 EC50 = 2500 nM T57943 CO0AG3 54583923 IC50 = 22.4 nM T57943 CI2DL4 54583924 EC50 = 1390 nM T57943 CV2WU1 54583925 IC50 = 13.4 nM T57943 CXA51D 54584867 IC50 = 11 nM T57943 C8YSL0 54585834 IC50 = 24.4 nM T57943 C9B5OF 54586343 IC50 = 26.9 nM T57943 C7A8ER 54587376 IC50 = 3.3 nM T57943 CE8T0H 54597799 IC50 = 2925 nM T57943 CFD30Q 56659222 IC50 = 29 nM T57943 CM64OW 56659923 IC50 = 24 nM T57943 C1NMH3 56659924 IC50 = 233 nM T57943 CR84YM 56661342 IC50 = 70 nM T57943 CUD26P 56663392 IC50 = 5125 nM T57943 CS3B4M 56663393 IC50 = 289 nM T57943 C8TZ9N 56666800 IC50 = 1075 nM T57943 CHW0D3 56666820 IC50 = 9300 nM T57943 CZO8E4 56666821 IC50 = 81500 nM T57943 COZ26R 56669572 IC50 = 15 nM T57943 C4J3TX 56670225 IC50 = 58600 nM T57943 C0BKU5 56670226 IC50 = 907 nM T57943 CD4QG1 56670255 IC50 = 22500 nM T57943 CH3Y9M 56670256 IC50 = 9920 nM T57943 CF38EO 56673751 IC50 = 7970 nM T57943 CW1R2X 56677088 IC50 = 10400 nM T57943 C8DN0E 56677089 IC50 = 4075 nM T57943 CUS83W 56678419 IC50 = 2600 nM T57943 C8MYW9 56679735 IC50 = 12 nM T57943 C8X7AY 56680385 IC50 = 3000 nM T57943 CB2R1I 56680416 IC50 = 2765 nM T57943 C72RGY 56683063 IC50 = 965 nM T57943 CKU26O 56683064 IC50 = 5533 nM T57943 C1U8MW 56683723 IC50 = 23000 nM T57943 C3FCG0 56683745 IC50 = 1410 nM T57943 C5O9SR 57333875 IC50 = 200000 nM T57943 CRC14J 59106264 IC50 = 13640 nM T57943 C64YGP 66572293 IC50 > 45000 nM T57943 CJU96E 66572295 IC50 > 45000 nM T57943 C49MTI 66572297 IC50 = 11320 nM T57943 C3U8QP 66572298 IC50 = 9760 nM T57943 CJ26SF 66572408 IC50 = 23740 nM T57943 C9Q7MU 66572409 IC50 = 25230 nM T57943 C6M5YT 66572411 IC50 = 10440 nM T57943 C74IMQ 66572412 IC50 = 24230 nM T57943 C43INL 66572413 IC50 = 10960 nM T57943 CRJ72C 66572414 IC50 = 8350 nM T57943 C6RK9I 66572520 IC50 = 9980 nM T57943 CZ59CH 66572521 IC50 = 7920 nM T57943 CCH08G 66572523 IC50 > 45000 nM T57943 CL7N3U 70683955 IC50 = 5270 nM T57943 CZTV25 70694451 IC50 = 15990 nM T57943 C1K5WF 70695295 IC50 > 80000 nM T57943 CGY3W2 71471109 IC50 = 30 nM T57943 CKZ2H0 71582971 IC50 = 349 nM T57943 C4WJ5F 71582972 IC50 = 94.3 nM T57943 CXA62J 71582973 IC50 = 92.3 nM T57943 CNZS31 71582974 IC50 = 1580 nM T57943 CE4L9D 71582975 IC50 = 170 nM T57943 CXMS80 71583078 IC50 = 184 nM T57943 C30UIL 71583079 IC50 = 1120 nM T57943 CJBC14 71583080 IC50 = 25.6 nM T57943 C57MOP 71583081 IC50 = 365 nM T57943 CS0YK9 71583082 IC50 = 346 nM T57943 C3UTO9 71583083 IC50 = 4.79 nM T57943 CW1R5Q 71583084 IC50 = 74.3 nM T57943 CR57LS 71583192 IC50 = 1060 nM T57943 C8B3NZ 71583193 IC50 = 46.8 nM T57943 CB6DY7 71583194 IC50 = 149 nM T57943 CHRZ40 71659499 IC50 = 4167 nM T57943 CG56UR 71659500 IC50 = 1167 nM T57943 CFED80 71659616 IC50 = 10710 nM T57943 CY38DX 71659617 IC50 = 8093 nM T57943 CF8J7Q 71659618 IC50 = 9628 nM T57943 CCO1Z2 71659619 IC50 = 3071 nM T57943 C5GYD7 71659620 IC50 = 16270 nM T57943 C0NZW9 71659621 IC50 = 438 nM T57943 C6W0MA 71659622 IC50 = 593 nM T57943 C4Y5CQ 71659623 IC50 = 9823 nM T57943 CAX05V 71659757 IC50 > 100000 nM T57943 C3LAV4 71659758 IC50 = 22050 nM T57943 CSZF46 71659759 IC50 = 85 nM T57943 C7O2JY 71659760 IC50 = 88 nM T57943 C4X0GI 71659761 IC50 = 74 nM T57943 C5L2KB 71659762 IC50 = 40 nM T57943 C4MQ8J 71659763 IC50 = 206 nM T57943 C6NO2V 71659764 IC50 = 241 nM T57943 C8AU2G 71659900 IC50 = 115 nM T57943 C7Q2ZN 71682003 IC50 = 187 nM T57943 CV96GT 71682004 IC50 = 106 nM T57943 C82YPX 71682161 IC50 = 25.9 nM T57943 CM76CD 71682162 IC50 = 23.3 nM T57943 CY07ID 71682310 IC50 = 56 nM T57943 CZI7D3 71682311 IC50 = 11.8 nM T57943 CJLY24 71698534 IC50 = 2570 nM T57943 CP3GS5 71698535 IC50 = 362 nM T57943 C6E5OV 71698716 IC50 > 500000 nM T57943 C9V4WS 71698717 IC50 > 500000 nM T57943 C26LVZ 71698718 IC50 > 500000 nM T57943 CAJ2N7 71698719 IC50 > 500000 nM T57943 C4CYG0 71698720 IC50 = 28500 nM T57943 C0ANH2 71698798 IC50 = 81100 nM T57943 C9O0CY 71698799 IC50 = 33400 nM T57943 C7CUJ8 71698800 IC50 = 42600 nM T57943 CIW75R 71698803 IC50 > 500000 nM T57943 C6EVI5 71698882 IC50 = 101000 nM T57943 CUM83A 71698883 IC50 = 18100 nM T57943 C2S7VN 71698884 IC50 = 16500 nM T57943 CP4Y9M 71698885 IC50 = 31800 nM T57943 CR4O3U 71698886 IC50 = 24500 nM T57943 CWDZ96 71698887 IC50 = 2390 nM T57943 CFP6Y2 71698973 IC50 = 1130 nM T57943 CIG39A 71698974 IC50 = 795 nM T57943 C25YSR 71698975 IC50 = 961 nM T57943 CG04WQ 71698976 IC50 > 500000 nM T57943 CR24DS 71698977 IC50 = 5990 nM T57943 C6PO1L 71698978 IC50 > 500000 nM T57943 CX1GO2 71699066 IC50 = 8840 nM T57943 CANH70 71716242 IC50 = 280 nM T57943 C40WIR 71718085 IC50 = 6500 nM T57943 CU75VK 71719897 IC50 = 6900 nM T57943 CBV6F1 71720507 IC50 > 100000 nM T57943 C8Y0GP 73345450 IC50 = 74 nM T57943 CGL6T9 73347421 IC50 > 500000 nM T57943 CBF89G 73353489 IC50 > 500000 nM T57943 CKYI28 73354985 IC50 > 500000 nM T57943 C7AM0E 76308407 IC50 = 181970085.9 nM T57943 CK67YV 76308408 IC50 = 123310483.3 nM T57943 CM3WU8 76308427 IC50 = 43954161.54 nM T57943 C4U5TO 76311196 IC50 = 12.8 nM T57943 CSI53E 76311200 IC50 = 7.1 nM T57943 CNOL37 76311201 IC50 = 9.6 nM T57943 C0ZBF1 76312084 IC50 = 157398286.5 nM T57943 C8IS5Q 76314800 IC50 = 3.1 nM T57943 CK41QI 76314804 IC50 = 11.6 nM T57943 CHS61N 76314805 IC50 = 13.7 nM T57943 C7U1DZ 76315606 IC50 = 215278173.5 nM T57943 CY0E6T 76315607 IC50 = 14996848.36 nM T57943 CMI3L9 76315608 IC50 = 359749335.2 nM T57943 CTS7X3 76315609 IC50 = 20989398.84 nM T57943 CDY7K0 76318413 IC50 = 8.1 nM T57943 CVPG02 76319292 IC50 = 15995580.29 nM T57943 C3EWP6 76319293 IC50 = 19998618.7 nM T57943 CB2N6G 76322078 IC50 = 2209 nM T57943 C8SPW6 76322082 IC50 = 15.2 nM T57943 C8I2FV 76322928 IC50 = 36982817.98 nM T57943 C4BFY2 76322948 IC50 = 3999447.5 nM T57943 CC2EP6 76325698 IC50 = 6.2 nM T57943 CZ02JB 76326490 IC50 = 926829823.4 nM T57943 CFD26R 76326504 IC50 = 23014418.17 nM T57943 C82YXK 76326505 IC50 = 54954087.39 nM T57943 CV9IN3 76326506 IC50 = 632411851.4 nM T57943 CL73GI 76330132 IC50 = 399944749.8 nM T57943 CMYR70 76330133 IC50 = 42953642.68 nM T57943 CPL76X 76330134 IC50 = 393550075.5 nM T57943 CH1VY9 76330152 IC50 = 26977394.32 nM T57943 CFY79U 76332916 IC50 = 6.3 nM T57943 CD35SI 76332917 IC50 = 4.4 nM T57943 C76IPD 76333770 IC50 = 460256573.6 nM T57943 CY16TU 76333771 IC50 = 33036954.1 nM T57943 CJFZ59 76333784 IC50 = 15995580.29 nM T57943 C5RXH6 76333785 IC50 = 15922087.27 nM T57943 CS59GO 76333786 IC50 = 209893988.4 nM T57943 C3FQX0 76336535 IC50 = 19.2 nM T57943 CV4PE6 76336536 IC50 = 13.9 nM T57943 CQ46DF 86279277 IC50 = 1.15 nM T57943 C0FDU4 86279278 IC50 = 56.85 nM T57943 C8QPA4 90654522 IC50 = 38.15 nM T57943 CI3UY0 90654523 IC50 = 41.53 nM T57943 CJ3DX6 90654524 IC50 = 49.39 nM T57943 C75MZK 90654525 IC50 = 80.55 nM T57943 CL2E7D 90654526 IC50 = 269.7 nM T57943 CMN74D 90654527 IC50 = 55.5 nM T57943 C2CUV9 90654528 IC50 = 13560 nM T57943 C3OC8I 90654529 IC50 = 180.8 nM T57943 C21PEL 90654530 IC50 = 62.01 nM T57943 CTFA68 90654531 IC50 = 97.92 nM T57943 CY63ON 90654532 IC50 = 22.1 nM T57943 CY8HP0 90654533 IC50 = 430.7 nM T57943 CHO1G0 90654534 IC50 = 783.4 nM T57943 COR17A 90654535 IC50 = 60.6 nM T57943 CLB31J 90654536 IC50 = 1270 nM T57943 C5Y6OL 90654537 IC50 = 1560 nM T57943 CP45YW 90654538 IC50 = 501 nM T57943 CB0YI1 90654539 IC50 = 729 nM T57943 CKCI60 90663142 IC50 = 512 nM T57943 C43QKY 101879103 IC50 = 34.9 nM T57943 CW02EX 101879104 IC50 = 49.7 nM T57943 C3SUH2 118723310 IC50 = 500000 nM T57943 C3M5TO 118723311 IC50 = 1190 nM T57943 CX82RL 118723312 IC50 = 210 nM T57943 C0SIK1 118723313 IC50 = 124 nM T57943 C3GPO7 118723314 IC50 = 17.4 nM T57943 C8H0EL 118723315 IC50 = 20.1 nM T57943 CTE1O2 118723316 IC50 = 50.7 nM T57943 CE8O9P 118723317 IC50 = 33.2 nM T57943 C3UZ6B 118723318 IC50 = 500000 nM T57943 C15RJF 118723319 IC50 = 353 nM T57943 C0OIE9 118723320 IC50 = 133 nM T57943 C01SDY 118723321 IC50 = 26.2 nM T57943 C0X9MJ 118723322 IC50 = 46.9 nM T57943 C5LB3W 118723323 IC50 = 81.4 nM T57943 C1GQO9 118723324 IC50 = 31.5 nM T57943 C48DEF 118723325 IC50 = 2.6 nM T57943 C67QMY 118723326 IC50 = 500000 nM T57943 CCJ27M 118723327 IC50 = 57.7 nM T57943 COG92V 118723328 IC50 = 4.8 nM T57943 CSX85P 118723329 IC50 = 500000 nM T57943 CICB42 118723330 IC50 = 2.9 nM T57943 C13BRQ 118723331 IC50 = 41 nM T57943 CDM0A7 118724007 IC50 = 292.1 nM T57943 CE01XH 118724008 IC50 = 199.9 nM T57943 C3MCW6 118724009 IC50 = 339.2 nM T57943 C9X0ZM 118724010 IC50 = 214.3 nM T57943 CNA7D6 118724011 IC50 = 218.6 nM T57943 CBWT97 118724012 IC50 = 548 nM T57943 CQA8U6 118724013 IC50 = 1344 nM T57943 C12EHA 118724014 IC50 = 185.7 nM T57943 CNB6M9 118724015 IC50 = 898.5 nM T57943 CL9AS6 118724016 IC50 = 1196 nM T57943 CX9D0V 118724017 IC50 = 192.6 nM T57943 CXT5V4 118724018 IC50 = 271.9 nM T57943 C6Q1IG 118724019 IC50 = 215.1 nM T57943 C59WMP 118724020 IC50 = 326.3 nM T57943 C7ZJL3 118724021 IC50 = 654.3 nM T57943 CG47EC 118724022 IC50 = 108.4 nM T57943 CJ6M2B 118724023 IC50 = 95 nM T57943 CNPQ61 118724024 IC50 = 119 nM T57943 CAWQ46 118724025 IC50 = 136.7 nM T57943 CM51UC 118724026 IC50 = 129.7 nM T57943 CO3J7G 118724027 IC50 = 87.7 nM T57943 CJ4F9Q 118724028 IC50 = 111.6 nM T57943 CN8A0V 118724029 IC50 = 47.3 nM T57943 C8TAO7 118724030 IC50 = 56.9 nM T57943 CP2QC1 118724031 IC50 = 181.6 nM T57943 CN5WS2 118724032 IC50 = 265.9 nM T57943 CXN5D4 118724033 IC50 = 389.7 nM T57943 CXZ70W 118724034 IC50 = 306.1 nM T57943 CQ68TB 118724035 IC50 = 32200 nM T57943 CJC7S1 118724036 IC50 = 235 nM T57943 CMN80F 118724037 IC50 = 126.6 nM T57943 CBNT42 118724038 IC50 = 140.6 nM T57943 C5S2MJ 118724039 IC50 = 264.6 nM T57943 CEB4O2 118724040 IC50 = 221.7 nM T57943 C9QKI3 127020966 IC50 = 75100 nM T57943 CV04JO 127037715 IC50 > 50000 nM T57943 CJ27CG 127042051 IC50 > 50000 nM T57943 CAT46D 127042341 IC50 > 50000 nM T57943 C6U1LV 132969040 IC50 = 60960 nM T57943 C45WQG 132969041 IC50 = 25080 nM T57943 CL6XW8 132969042 IC50 = 29260 nM T57943 CWM2E8 133081971 IC50 > 9999 nM T57943 C51HUD 134140107 IC50 = 44740 nM T57943 C0S6OI 134142875 IC50 = 51490 nM T57943 C9A2GK 134156912 IC50 > 100000 nM T57943 CU79RM 135402730 Ki = 310 nM T57943 CB68PL 135402731 Ki = 400 nM T57943 C4DXF1 135444600 IC50 = 0.8 ug.mL-1 T57943 CH9YR2 135501892 EC50 = 430 nM T57943 CJ1HI2 135532687 IC50 = 0.02 ug.mL-1 T57943 C0LUX4 135533972 EC50 > 50000 nM T57943 C2IG7M 135559049 Ki = 500 nM T57943 C3NGY4 135559050 Ki = 100 nM T57943 CQ2BG5 137007045 EC50 = 18230 nM T57943 C54QCM 137083623 EC50 = 1420 nM T57943 CT65FY 137083624 EC50 = 4960 nM T57943 CJ8VA9 137083625 EC50 = 2420 nM T57943 CXF5H6 137083626 EC50 = 4260 nM T57943 CM7W2N 137083627 EC50 = 250 nM T57943 CLDI36 137225012 IC50 = 487200 nM T57943 C17RCJ 137225013 IC50 = 547000 nM T57943 C4H1LQ 137225014 IC50 = 551500 nM T57943 C0J4OC 137225015 IC50 = 598600 nM T57943 COR46U 137225016 IC50 = 375300 nM T57943 C2LDY7 137225026 IC50 = 674300 nM T57943 CK7A2F 137225027 IC50 = 310000 nM T57943 C0PO9W 137225044 IC50 = 63200 nM T57943 CIFN92 137225052 IC50 = 350600 nM T57943 C73PVR 137225053 IC50 = 121700 nM T57943 CGXB30 137225054 IC50 = 129500 nM T57943 C2DFG6 137225055 IC50 = 132400 nM T57943 CW41CO 137225056 IC50 = 19400 nM T57943 CH26XP 137225057 IC50 = 35000 nM T57943 C7TE5N 137225058 IC50 = 38300 nM T57943 CM2P1A 137225080 IC50 = 456100 nM T57943 C5FIE7 137225081 IC50 = 202400 nM T57943 CZX0Y5 137225082 IC50 = 278200 nM T57943 C7D4QS 137225083 IC50 = 296500 nM T57943 C9TK5D 137225091 IC50 = 52340 nM T57943 C7UFH6 137225092 IC50 = 37200 nM T57943 CA6EI9 138480034 IC50 = 138 nM T57943 CM0NI2 138480059 IC50 = 14 nM T57943 CSH5X3 138480060 IC50 = 10 nM T57943 CE10UI 138480076 IC50 = 30 nM T57943 CT1Y6G 138480108 IC50 = 20 nM T57943 CY0G3A 138480119 IC50 = 108 nM T57943 C1V6LD 138480124 IC50 = 79 nM T57943 CL8NG5 138480135 IC50 = 25 nM T57943 CZEY23 138480158 IC50 = 14 nM T57943 C9IR7C 138480171 IC50 = 6 nM T57943 CP1BN5 138480172 IC50 = 30 nM T57943 C9TV2K 138480174 IC50 = 112 nM T57943 C9CV0K 138480175 IC50 = 27 nM T57943 CR3XZ4 138480178 IC50 = 9 nM T57943 C2Y9IX 138480200 IC50 = 142 nM T57943 CUY9X6 138480234 IC50 = 40 nM T57943 CT5S0A 138480241 IC50 = 14 nM T57943 CGX82L 138480283 IC50 = 26 nM T57943 C3GWL5 138480291 IC50 = 18 nM T57943 CYKQ07 138480294 IC50 = 20 nM T57943 CA2TZ4 138480315 IC50 = 142 nM T57943 CN68PV 138480326 IC50 = 18 nM T57943 C3HX6C 138480330 IC50 = 12 nM T57943 CHX2Q5 138480333 IC50 = 6 nM T57943 C0EG8A 138480341 IC50 = 20 nM T57943 C4OHT6 138480455 IC50 = 27 nM T57943 CTS58J 138480477 IC50 = 14 nM T57943 CN6C5O 138480509 IC50 = 6 nM T57943 C65DQG 138480529 IC50 = 24 nM T57943 C8SB7X 138480537 IC50 = 10 nM T57943 CAZ2L4 138616824 IC50 = 64 nM T57943 C4YFG8 138616827 IC50 = 21 nM T57943 C8PKO6 138616828 IC50 = 213 nM T57943 C48GMN 138617058 IC50 = 44 nM T57943 C1SZ4A 138617074 IC50 = 7 nM T57943 CJHR93 138617075 IC50 = 19 nM T57943 CWL24C 145967811 IC50 = 244 nM T57943 CP4LR5 145967828 IC50 = 35 nM T57943 CQX2J4 145968113 IC50 = 75 nM T57943 CDN6P4 145968607 IC50 = 20 nM T57943 CQNH57 145968735 IC50 = 12 nM T57943 C0SEQ8 145969321 IC50 = 23 nM T57943 CHLR92 145969539 IC50 = 22 nM T57943 C87GLY 145969570 IC50 = 16 nM T57943 C05NAY 145988824 IC50 = 11 nM T57943 CW1Q0T 155525619 IC50 = 7600 nM T57943 CU42CE 155567829 IC50 > 100000 nM T57943 D01XMM 4117383 IC50 = 2197.86 nM T57943 D05GGE 11652039 IC50 = 544 nM T57943 D09AED 11357566 IC50 = 331 nM T57943 D09GKA 11522185 IC50 = 4630 nM T57943 D0B6VI 9903426 IC50 = 169.82 nM T57943 D0B8HU 11629882 IC50 = 261 nM T57943 D0D4RW 9839586 IC50 = 1900 nM T57943 D0FZ7W 1714901 IC50 = 255 nM T57943 D0G2DQ 4669250 IC50 = 1000 nM T57943 D0IQ7Y 935415 IC50 = 465.7 nM T57943 D0L3PO 11680763 IC50 = 630 nM T57943 D0L9AX 644345 IC50 = 0.2 nM T57943 D0N5MU 4117381 Ki = 1400 nM T57943 D0N6BC 950368 Ki = 100000 nM T57943 D0Q9XX 515950 Ki = 500 nM T57943 D0SP2O 7054 IC50 > 100000 nM T57943 D0U3JD 16358 IC50 > 50000 nM T57943 D0V6DX 10640 IC50 = 149 nM T57943 D0Y5IQ 44255320 IC50 = 5000 nM T57943 D0Y7HC 44310146 Ki = 26 nM T00749 C3VRO9 44557921 IC50 > 10000 nM T00749 CV63UL 67240318 IC50 > 10000 nM T00749 CUW38G 137297825 IC50 < 50 nM T00749 C2YOP9 137297852 IC50 < 50 nM T00749 C2MD1Q 155513187 IC50 > 10000 nM T00749 D0M5FF 5083 IC50 = 52.9 nM T95295 CG5B6C 153054 IC50 > 500000 nM T95295 C9VCM0 514258 IC50 > 125000 nM T95295 CCRW58 514263 IC50 = 125000 nM T95295 C0L2TF 23725128 IC50 > 500000 nM T60631 D01PZD 5329098 IC50 = 170 nM T60631 D03ZBT 11626560 IC50 > 10000 nM T60631 D04LVK 57379345 IC50 = 2304 nM T60631 D09KTS 24821094 IC50 = 5.2 nM T60631 D09XZB 123631 IC50 = 1700 nM T60631 D0E6XR 3062316 IC50 = 433 nM T60631 D0G6QF 3081361 IC50 = 49 nM T60631 D0H0EQ 24826799 IC50 = 0.3 nM T60631 D0IQ6P 25102847 IC50 = 2.4 nM T60631 D0K8KX 5280343 IC50 = 78100 nM T60631 D0R0FO 9823820 Ki = 1.5 nM T60631 D0R0MW 5329102 IC50 < 1 nM T60631 D0U3SY 49806720 IC50 = 4.8 nM T60631 D0W5HK 216239 IC50 = 6 nM T60631 D00DRL 44137946 IC50 = 640 nM T60631 D02RJY 11442891 IC50 = 31 nM T60631 D03HUX 49792852 IC50 > 10000 nM T60631 D03LWG 53235510 IC50 = 3352 nM T60631 D05PZB 135398495 IC50 = 1 nM T60631 D06KTJ 53252276 IC50 = 8.4 nM T60631 D07EHV 44814409 IC50 > 10000 nM T60631 D07HPJ 11476171 IC50 = 3300 nM T60631 D08HOM 46207586 IC50 = 7 nM T60631 D0AX4H 78427026 IC50 = 0.4 nM T60631 D0E3TC 44259 IC50 = 1.69 nM T60631 D0FD6D 11751922 IC50 = 5 nM T60631 D0G2QH 10297043 IC50 = 740 nM T60631 D0G8BM 16722836 IC50 = 48 nM T60631 D0G9AW 59473233 EC50 > 1000 nM T60631 D0M9QZ 11485656 IC50 = 1900 nM T60631 D0O0LS 25141092 IC50 = 393 nM T60631 D0O6WV 24794418 IC50 = 594 nM T60631 D0P1CV 46191454 IC50 > 10000 nM T60631 D0Q9UX 16718576 IC50 = 1933 nM T60631 D0S6TK 11213558 EC50 = 36 nM T60631 D0S7HM 16041424 IC50 = 10 nM T60631 D0T2ER 24767976 IC50 = 18 nM T60631 D0Z4RC 24756910 IC50 = 3200 nM T60631 D03BNU 59604787 IC50 > 10000 nM T60631 D00DQX 11667893 IC50 = 90 nM T60631 D01MIP 6536806 IC50 = 1000 nM T60631 D0T3ME 156422 IC50 = 30 nM T60631 CB1VW3 1400 IC50 = 11 nM T60631 C8HN2C 3798 IC50 = 1700 nM T60631 CO6B3I 265711 IC50 = 20900 nM T60631 C1ZG2U 449087 IC50 > 10000 nM T60631 CYB5E2 1749976 IC50 = 170 nM T60631 C1RQ4E 1886699 IC50 = 4800 nM T60631 C6NK9W 1898760 IC50 = 1600 nM T60631 C8S0UP 2806990 IC50 = 9380 nM T60631 C2AFE3 2808988 IC50 = 1200 nM T60631 C9Z1FJ 2810885 IC50 = 54000 nM T60631 CH4V8I 2811823 IC50 = 6160 nM T60631 CH64KM 2814387 IC50 = 82600 nM T60631 CI6VH2 2817227 IC50 = 12100 nM T60631 COV8U0 2817495 IC50 = 6470 nM T60631 C2FO4B 5329010 IC50 = 0.75 nM T60631 C2O9ZG 5391486 IC50 = 68400 nM T60631 CCT39K 5703472 IC50 = 9400 nM T60631 CQ3S8L 6450842 IC50 > 100000 nM T60631 CTAI98 9839842 IC50 = 45000 nM T60631 CD17IK 9869078 IC50 = 6 nM T60631 CX23IZ 9926213 IC50 = 1600 nM T60631 CTQ48P 9927432 IC50 = 3 nM T60631 CUJR40 10062694 EC50 = 77 nM T60631 C7SFI1 10296883 IC50 > 10000 nM T60631 CY9F3G 10425574 IC50 = 4.6 nM T60631 C7HBP6 10429593 IC50 > 10000 nM T60631 C6AJI9 10562777 IC50 = 8000 nM T60631 CM8N6L 10593765 IC50 = 3700 nM T60631 C9Z7XH 10663503 IC50 = 100000 nM T60631 CACS26 11561968 Ki > 2000 nM T60631 C51SLY 11645208 IC50 = 100000 nM T60631 CU0E8O 11690457 Ki > 2000 nM T60631 C2GCB7 11779327 IC50 = 590 nM T60631 CUE65C 11818023 IC50 = 4100 nM T60631 C9JT4S 11847343 IC50 = 113 nM T60631 CQN23V 15551239 IC50 = 300 nM T60631 CQG45C 16109001 IC50 = 8300 nM T60631 C5VPH9 16129448 IC50 = 132 nM T60631 CV7Q2B 16876702 IC50 = 280 nM T60631 CSK5L4 18770844 IC50 = 600 nM T60631 C60QKI 21260292 IC50 = 23 nM T60631 CUH32C 21260305 IC50 = 0.41 nM T60631 CA51HY 21701560 IC50 = 10 nM T60631 CVI49J 21701562 IC50 = 100 nM T60631 C3VT6O 21701572 IC50 = 1.1 nM T60631 CDS7B0 22172654 IC50 = 2900 nM T60631 C6G4JM 22172657 IC50 = 3.9 nM T60631 C2V9BG 22394608 IC50 = 7500 nM T60631 C3F9LN 23366726 IC50 = 1700 nM T60631 C4QU3A 23366752 IC50 = 140 nM T60631 CR3M1N 23644582 IC50 = 25 nM T60631 CRF4T1 23646049 IC50 = 100000 nM T60631 C5W1PI 23646055 IC50 = 10000 nM T60631 C7RJ3O 23646063 IC50 = 100000 nM T60631 CXC16Y 23646065 IC50 = 1000 nM T60631 CX3H1O 23647607 IC50 = 66000 nM T60631 CBD9U4 23647620 IC50 = 460 nM T60631 C1Z3GO 23655831 IC50 = 200 nM T60631 CAJ4T2 24762205 IC50 = 4700 nM T60631 CQNP54 24764449 IC50 = 25000 nM T60631 CQN3Z7 24825710 IC50 = 614 nM T60631 C70FVX 24860829 IC50 = 128 nM T60631 C5TPL9 24866033 IC50 = 290 nM T60631 CD40VG 24866217 IC50 = 130 nM T60631 C43HWQ 24883287 IC50 = 700 nM T60631 C8DA5Q 24883334 IC50 < 100 nM T60631 CD5V2B 24951139 IC50 = 250 nM T60631 C4EG8R 24993189 IC50 > 10000 nM T60631 CFT5S4 24994207 IC50 = 91 nM T60631 CJ2HX8 25023824 IC50 = 100 nM T60631 CRTY12 25023826 IC50 = 75 nM T60631 C9Z0AL 25023827 IC50 = 25 nM T60631 CX30ZW 25023828 IC50 = 75 nM T60631 C0Q7KX 25023829 IC50 = 6 nM T60631 CI7ZE2 25023830 IC50 = 80 nM T60631 CVD53O 25023831 IC50 = 95 nM T60631 CIVA70 25023832 IC50 = 90 nM T60631 COD9G1 25023833 IC50 = 85 nM T60631 CM4CF6 25023834 IC50 = 34 nM T60631 C6SC3L 25023835 IC50 > 1000 nM T60631 CSDU50 25060093 IC50 = 2000 nM T60631 C4KJ3F 25147774 IC50 = 110 nM T60631 CIZ6F1 25147782 IC50 = 60 nM T60631 CNG96H 25210579 IC50 > 10000 nM T60631 CNQ9G5 25218180 IC50 < 1000 nM T60631 CCFQ29 44187005 IC50 = 160 nM T60631 CN8WB9 44189332 IC50 = 15 nM T60631 C4JH9V 44415997 IC50 = 3721 nM T60631 CEOG74 44416018 IC50 = 337 nM T60631 C6UR0Y 44416036 IC50 = 100000 nM T60631 CKN4Z2 44416037 IC50 = 10000 nM T60631 C2R8HM 44416063 IC50 = 10000 nM T60631 CF83LU 44416088 IC50 = 10000 nM T60631 CFR9H4 44416107 IC50 = 1000 nM T60631 C9ZLI1 44416137 IC50 = 1000 nM T60631 CY3DC8 44433305 IC50 > 1000 nM T60631 C9RP8G 44440760 IC50 = 50 nM T60631 C6G5RH 44440761 IC50 = 580 nM T60631 CMR72W 44440766 IC50 > 3000 nM T60631 CK6V1L 44511478 IC50 = 9204 nM T60631 CHX67O 44512175 IC50 = 4246 nM T60631 CO3B5L 44512176 IC50 = 1800 nM T60631 C3VRO9 44557921 IC50 > 10000 nM T60631 CN46LW 44563276 IC50 = 480 nM T60631 CAQ47L 44563277 IC50 = 600 nM T60631 CO4Y1W 44563313 IC50 > 600 nM T60631 C15AJI 44563338 IC50 > 600 nM T60631 CDG27P 44563339 IC50 = 90 nM T60631 CU3RF1 45139989 IC50 > 10000 nM T60631 CQGZ06 45139991 IC50 > 10000 nM T60631 CF57GK 46215462 IC50 = 3 nM T60631 C2P9QO 46228508 IC50 = 698 nM T60631 C6E5PY 46228822 IC50 = 202 nM T60631 C3T8AM 46228951 IC50 = 237 nM T60631 C6S1RT 46233106 IC50 = 20000 nM T60631 C7JM9T 46233107 IC50 = 1100 nM T60631 C85RJI 46233108 IC50 = 580 nM T60631 CO1KJ2 46233109 IC50 = 12000 nM T60631 CSL52F 46233110 IC50 = 78000 nM T60631 CNE60M 46233143 IC50 = 63000 nM T60631 CB3CT4 46233145 IC50 = 1000 nM T60631 COBF49 46233146 IC50 = 66000 nM T60631 CTCO76 46233147 IC50 = 34000 nM T60631 CUI46Q 46233183 IC50 = 5900 nM T60631 C5CH1F 46233184 IC50 = 23000 nM T60631 C19SZF 46233185 IC50 = 210 nM T60631 C7ON5A 46233287 IC50 > 10000 nM T60631 CJB06K 46233299 IC50 = 1700 nM T60631 CL98DY 46233648 IC50 = 2000 nM T60631 CWPS75 46233680 IC50 = 5500 nM T60631 CMV56B 46233681 IC50 = 1400 nM T60631 C1PS3B 46233682 IC50 = 22000 nM T60631 CNH29U 46233683 IC50 = 40000 nM T60631 C21NWZ 46838816 IC50 = 8000 nM T60631 CJ61LQ 46838817 IC50 = 10000 nM T60631 CL07DO 46838818 IC50 = 2300 nM T60631 C26HDB 46838819 IC50 = 8600 nM T60631 C6WC8N 46838820 IC50 = 14000 nM T60631 C6LWY5 46838821 IC50 = 27000 nM T60631 CWD7M9 46838822 IC50 = 19000 nM T60631 CH7Z8X 46838962 IC50 = 8300 nM T60631 CYKJ29 46838963 IC50 = 13000 nM T60631 CQE01F 46838964 IC50 = 11000 nM T60631 C0TL7Y 46838965 IC50 = 9200 nM T60631 CNW6I7 46838966 IC50 = 3400 nM T60631 C9DR6V 46838967 IC50 = 690 nM T60631 C4O2BK 46838968 IC50 = 3600 nM T60631 C8BR0O 46839102 IC50 = 5000 nM T60631 C5OCP1 46839103 IC50 = 39000 nM T60631 C6KBQ3 46839104 IC50 = 3600 nM T60631 CL82BU 46839105 IC50 = 26000 nM T60631 CLS29B 46872626 IC50 > 10000 nM T60631 CRA74I 49842779 IC50 > 10000 nM T60631 CF91RS 49843531 IC50 > 10000 nM T60631 C2Y6QS 50938552 IC50 > 10000 nM T60631 C61DVY 50990961 IC50 = 1.6 nM T60631 CV3UP9 50992247 IC50 = 0.8 nM T60631 CS9G6E 50997096 IC50 > 10000 nM T60631 C9NYP4 51036677 IC50 > 10000 nM T60631 C4WRY3 51037112 IC50 > 10000 nM T60631 CRI28Z 51037948 IC50 > 10000 nM T60631 CEQN27 52936621 Ki > 1000 nM T60631 C09SDH 53257410 IC50 > 10000 nM T60631 CZ0BV7 53320342 IC50 > 10000 nM T60631 C2W9OA 53324451 IC50 = 7200 nM T60631 CBK9Q6 53357848 IC50 > 10000 nM T60631 C8NA4L 53384644 IC50 = 3700 nM T60631 CE1ZK6 54759168 IC50 > 10000 nM T60631 C8AB1J 54759606 Ki = 18 nM T60631 CM8JX1 56604907 IC50 = 10 nM T60631 C0EXV7 56659745 IC50 = 484 nM T60631 CHDT04 56659827 IC50 = 100000 nM T60631 C84VHN 56663232 IC50 = 10000 nM T60631 CELF89 56663293 IC50 = 500 nM T60631 C7WXI0 56663294 IC50 = 1600 nM T60631 CUG58E 56663295 IC50 = 1800 nM T60631 C1X4HT 56666656 IC50 = 212 nM T60631 CGO6Z7 56666657 IC50 = 692 nM T60631 CW38SB 56670084 IC50 = 1117 nM T60631 C85QPF 56670142 IC50 = 100000 nM T60631 C5GOX1 56673427 IC50 = 10000 nM T60631 CXAZ93 56673428 IC50 = 90 nM T60631 C9IK8M 56673513 IC50 = 10000 nM T60631 CF7YH2 56676920 IC50 = 753 nM T60631 CKV7O4 56676921 IC50 = 1232 nM T60631 C6QU9Y 56676979 IC50 = 4500 nM T60631 C64QPN 56676980 IC50 = 11000 nM T60631 C0C7UK 56680225 IC50 = 537 nM T60631 CM83DX 56680234 IC50 = 1262 nM T60631 CTUJ32 56680305 IC50 = 55000 nM T60631 C18LIP 56680320 IC50 = 110 nM T60631 CP2OY0 56683628 IC50 = 2700 nM T60631 CI6QE5 56970263 IC50 < 500 nM T60631 C62OJE 56970264 IC50 = 66 nM T60631 CZSM95 57412684 IC50 > 10000 nM T60631 C8QVX0 57523390 IC50 = 50 nM T60631 CF3HI1 57523419 IC50 = 110 nM T60631 C3YP6K 57523420 IC50 = 195 nM T60631 C84XWL 57523425 IC50 = 83 nM T60631 CI50KU 58167984 IC50 = 706 nM T60631 CP34RY 59394193 IC50 = 500 nM T60631 CB5I1N 59662500 IC50 = 4300 nM T60631 C1MR8Q 60097495 IC50 > 1000 nM T60631 C9ZCT2 62705065 IC50 > 1000 nM T60631 CD2BZ5 66549796 IC50 = 8 nM T60631 C10AMI 66553589 IC50 = 210 nM T60631 C1HSE0 67035086 IC50 = 8 nM T60631 CWI6K5 67035106 IC50 > 10000 nM T60631 C38RGB 67035556 IC50 = 4400 nM T60631 CV3HW2 67035568 IC50 = 970 nM T60631 C37NKO 67129970 IC50 = 3500 nM T60631 CK80LJ 67130050 IC50 = 2950 nM T60631 CV63UL 67240318 IC50 > 10000 nM T60631 C8I7GC 68293638 IC50 = 6000 nM T60631 CD56XK 68293660 IC50 = 9300 nM T60631 C7GRV2 68755406 IC50 = 1510 nM T60631 CM9RU2 69519173 IC50 = 29 nM T60631 C7VJ6A 70647728 IC50 = 110 nM T60631 CN32CE 70686389 IC50 = 43 nM T60631 CAW17X 71494057 IC50 > 25000 nM T60631 CDE4X6 71494225 IC50 > 25000 nM T60631 CCN01X 71547862 IC50 > 10000 nM T60631 C1BCX0 71579696 IC50 > 1000 nM T60631 CS62NH 71698376 IC50 = 67.8 nM T60631 C3OS8U 71714087 IC50 = 4 nM T60631 C92AZQ 71714088 IC50 = 54 nM T60631 CN1Y9I 71714230 IC50 = 75 nM T60631 CM6NE9 71714231 IC50 = 6 nM T60631 CG28AP 71714232 IC50 = 25 nM T60631 C91CRY 71714233 IC50 = 34 nM T60631 C67HDT 71714234 IC50 = 140 nM T60631 CRS05F 71714235 IC50 = 5 nM T60631 CVC19T 71714373 IC50 = 25 nM T60631 CD5C8J 71714374 IC50 = 150 nM T60631 C51ISR 71714375 IC50 = 300 nM T60631 C5HJK2 71714376 IC50 = 4 nM T60631 C70SJV 71714377 IC50 = 73 nM T60631 C59UBD 71716995 IC50 > 30000 nM T60631 C60TUV 72737208 IC50 = 223 nM T60631 CJ3WA6 72737404 IC50 = 347 nM T60631 C2PAK9 73438493 IC50 = 1 nM T60631 CGDB30 74538658 IC50 = 10 nM T60631 CBAT06 76071144 IC50 = 7 nM T60631 C2O6TS 76311163 IC50 = 5470 nM T60631 CI8H9X 76311164 IC50 = 57200 nM T60631 CVU96Q 76311165 IC50 = 7040 nM T60631 C9RDO6 76314767 IC50 = 12850 nM T60631 C3I7UA 76314769 IC50 = 9070 nM T60631 CRO31B 76318365 IC50 = 58600 nM T60631 CA95JI 76318366 IC50 = 9640 nM T60631 CGYM87 76318367 IC50 = 24100 nM T60631 C8JRL6 76322049 IC50 = 7960 nM T60631 C25ORT 76325670 IC50 = 17100 nM T60631 C38HPS 76329233 IC50 = 22400 nM T60631 CB5RH9 76329234 IC50 = 4260 nM T60631 C9J6FO 76329235 IC50 = 28100 nM T60631 CN18KC 76329236 IC50 = 9260 nM T60631 C9PDY0 76332896 IC50 = 15300 nM T60631 C2JUZ1 76332897 IC50 = 10300 nM T60631 CT84NC 76336503 IC50 = 7900 nM T60631 C4SQ2V 76336505 IC50 = 22600 nM T60631 C5U8VI 78426332 IC50 = 0.4 nM T60631 C7SPD9 78426333 IC50 <= 100 nM T60631 CE9R4L 78426885 IC50 = 0.4 nM T60631 CN0X2A 78427023 IC50 = 0.4 nM T60631 C4VUP1 78427168 IC50 = 1.7 nM T60631 CCJ43A 86302281 IC50 = 1626 nM T60631 CB5NJ4 86302541 IC50 = 20.2 nM T60631 CPG3A5 86302574 IC50 > 30000 nM T60631 CS7GX8 89708625 IC50 = 9594 nM T60631 CY0UC4 90645194 IC50 > 10000 nM T60631 CX29IY 90655145 IC50 > 10000 nM T60631 CPGV73 101884319 IC50 = 56 nM T60631 CA1TZ3 101884321 IC50 = 140 nM T60631 CG9KE7 101884322 IC50 = 120 nM T60631 C84MVD 101884325 IC50 = 330 nM T60631 CV9S8Q 118111994 IC50 = 24 nM T60631 C5QW0Y 118111995 IC50 = 100 nM T60631 CH6M2V 118112005 IC50 = 10 nM T60631 CRL0O1 118112011 IC50 = 190 nM T60631 CGI47W 118112014 IC50 = 9.3 nM T60631 CU25TZ 118112016 IC50 = 23 nM T60631 C4QB8Y 118112024 IC50 = 38 nM T60631 C0KO2J 118112026 IC50 = 130 nM T60631 CHCI59 118112037 IC50 = 350 nM T60631 CAD76E 118112040 IC50 = 2 nM T60631 CWU3S7 118112047 IC50 = 19 nM T60631 C29BPV 118112051 IC50 = 14 nM T60631 CS06EV 118112055 IC50 = 1100 nM T60631 C4VBY7 118112056 IC50 = 3800 nM T60631 CYEO57 118112076 IC50 = 1.7 nM T60631 C8AE2F 118112077 IC50 = 44 nM T60631 CD61JA 118112079 IC50 = 30 nM T60631 CBA4O8 118112080 IC50 = 29 nM T60631 CM1E5A 118112082 IC50 = 15 nM T60631 CJ94NF 118112083 IC50 = 5500 nM T60631 C2AQ6Y 118112087 IC50 = 15 nM T60631 C5QAZ7 118112091 IC50 = 120 nM T60631 CNO0T7 118112099 IC50 = 48 nM T60631 CH84RT 118112100 IC50 = 17 nM T60631 CU6MI0 118112101 IC50 = 11 nM T60631 C02OVL 118112108 IC50 = 44 nM T60631 C7ACP6 118112114 IC50 = 3.9 nM T60631 C5FT9N 118112115 IC50 = 12 nM T60631 C4B1FL 118112118 IC50 = 5 nM T60631 CT6A1B 118112122 IC50 = 14 nM T60631 CTK8O1 118112125 IC50 = 100 nM T60631 C0S9QW 118112133 IC50 = 78 nM T60631 C0SQ7Y 118112144 IC50 = 23 nM T60631 CR58UD 118112154 IC50 = 21 nM T60631 CO3WA5 118112158 IC50 = 7 nM T60631 C23GBT 118112186 IC50 = 4.8 nM T60631 C5HB0N 118112191 IC50 = 120 nM T60631 CE9ZN0 118112194 IC50 = 18 nM T60631 COD73Q 118112202 IC50 = 62 nM T60631 CU02NF 118559124 IC50 = 1.6 nM T60631 CY7BI2 118706214 IC50 > 10000 nM T60631 CBV46P 118712373 IC50 > 100000 nM T60631 CKD7X1 118712374 IC50 > 100000 nM T60631 C3OJP1 118712375 IC50 > 100000 nM T60631 CI3C7E 118712376 IC50 = 67800 nM T60631 C8Y7TM 118712377 IC50 = 18800 nM T60631 C5TOA1 118712378 IC50 = 15700 nM T60631 CE2O3J 118712379 IC50 = 210 nM T60631 CV4N7Z 118712380 IC50 = 22300 nM T60631 CDFZ85 118712381 IC50 = 20400 nM T60631 CK05BQ 118712382 IC50 = 19300 nM T60631 C7N1AF 118712383 IC50 = 17200 nM T60631 CA4VN0 118712384 IC50 = 14300 nM T60631 CT8Y9Q 118712385 IC50 = 9100 nM T60631 CC2FT8 118712386 IC50 = 2500 nM T60631 CKBP72 121231408 IC50 > 10000 nM T60631 C81IFQ 122163152 IC50 > 100000 nM T60631 C08KEM 122179540 IC50 = 4900 nM T60631 C3AJ4C 122179546 IC50 = 8000 nM T60631 CG0RP7 122179547 IC50 = 3700 nM T60631 C1A0SQ 122179548 IC50 = 6000 nM T60631 CB0QF4 122183083 IC50 = 210 nM T60631 CB2VY7 122183099 IC50 = 63 nM T60631 CZ1U4R 122183100 IC50 = 64 nM T60631 C4X7SD 122192466 IC50 = 986 nM T60631 C8YA0F 122628813 IC50 = 2.6 nM T60631 COC02I 122629035 IC50 = 8.4 nM T60631 CD67LU 122705248 IC50 = 289 nM T60631 CX63VW 122705258 IC50 > 10000 nM T60631 C76IKM 122705261 IC50 = 598 nM T60631 CY30FL 123752658 IC50 = 1.3 nM T60631 C8ALO2 124088839 IC50 > 10000 nM T60631 CP4G1B 126591726 IC50 = 96 nM T60631 C8AF6C 126591906 IC50 = 41 nM T60631 C08MPD 126591909 IC50 = 910 nM T60631 C9N6BO 126591918 IC50 = 68 nM T60631 CW0C1U 126591922 IC50 = 2 nM T60631 C2LAM7 126591927 IC50 = 3 nM T60631 CRC78F 126592010 IC50 = 241 nM T60631 C9MRH4 126592018 IC50 = 150 nM T60631 C5E6MK 126592021 IC50 = 241 nM T60631 CJQ40U 126592025 IC50 = 74 nM T60631 C6RX2P 126592026 IC50 = 213 nM T60631 C6YUX2 126592031 IC50 = 190 nM T60631 CFB82J 126592038 IC50 = 583 nM T60631 CHZ0G6 126592040 IC50 = 910 nM T60631 CZ1R2Q 126592042 IC50 = 52 nM T60631 CD16GH 126592159 IC50 = 2100 nM T60631 C4F1EX 126592165 IC50 = 27 nM T60631 CFS64Y 126592360 IC50 = 5 nM T60631 CT15BX 126592367 IC50 = 41 nM T60631 CB3J5F 127030529 IC50 = 9.7 nM T60631 C2U0HN 127031755 IC50 = 5 nM T60631 CR5M3P 127032029 IC50 = 13 nM T60631 C83CIL 127032326 IC50 = 4100 nM T60631 CSG9N6 127033539 IC50 = 11 nM T60631 CES05I 127033845 IC50 > 10000 nM T60631 CH23IT 127033855 IC50 = 3.2 nM T60631 CVX2W5 127033856 IC50 = 2.6 nM T60631 C6SV1L 127034132 IC50 = 210 nM T60631 CL5KS6 127034133 IC50 = 16 nM T60631 CY4SV3 127034402 IC50 = 60 nM T60631 CKS28E 127034802 IC50 = 1.6 nM T60631 C13TVG 127036442 IC50 = 8330 nM T60631 CZD87E 127037084 IC50 = 3 nM T60631 CKX40V 127037812 IC50 = 167.1 nM T60631 C70RUP 127038480 IC50 = 59.2 nM T60631 CB9Z0V 127038973 IC50 = 2 nM T60631 C3WCN8 127041777 IC50 = 22.8 nM T60631 CG8DA9 127045861 IC50 > 100000 nM T60631 CHK16Q 127045929 IC50 > 1000 nM T60631 CMD1Y6 127046108 IC50 = 14 nM T60631 CD4G0C 127046310 IC50 = 9 nM T60631 CI8HJ2 127046833 IC50 = 4300 nM T60631 CC4ND8 127046862 IC50 > 100000 nM T60631 C5KX9R 127046975 IC50 = 65 nM T60631 CT0SU2 127046976 IC50 = 11 nM T60631 CY3J0C 127047591 IC50 > 1000 nM T60631 CLB09X 127047634 IC50 = 3300 nM T60631 CL8GM6 127047677 IC50 = 7700 nM T60631 CQPV90 127047678 IC50 = 9100 nM T60631 CHTS05 127047813 IC50 = 150 nM T60631 C6B1MP 127047814 IC50 = 110 nM T60631 CO25WH 127052538 IC50 = 6584 nM T60631 CT06ZP 132008468 IC50 = 1.2 nM T60631 C96WRI 132008498 IC50 = 0.1 nM T60631 CUO0C5 132156633 IC50 > 10000 nM T60631 C6OMB1 132204257 IC50 = 32 nM T60631 CJ04HZ 132585195 IC50 > 1000 nM T60631 CERS64 132937256 IC50 > 30000 nM T60631 CDT95V 134135856 IC50 = 1.8 nM T60631 CR1YW6 134141181 IC50 = 21.4 nM T60631 CL0HJ2 134142263 IC50 = 137.8 nM T60631 C3OHY7 134142284 IC50 = 2.5 nM T60631 CMQA15 134143603 IC50 = 26.6 nM T60631 CQ8I9E 134144809 IC50 = 19.4 nM T60631 CUKH90 134146405 IC50 = 17.9 nM T60631 C2JX3Y 134147460 IC50 = 2.1 nM T60631 CI79OS 134153552 IC50 = 107.6 nM T60631 C8B4NA 134154798 IC50 = 7.3 nM T60631 C7WO8J 134155588 IC50 = 341.9 nM T60631 CP2TX7 134156446 IC50 = 11.4 nM T60631 CLO25D 134157865 IC50 = 12.4 nM T60631 CIK38Q 134229735 IC50 = 71.6 nM T60631 CYL5V1 134694986 IC50 > 30000 nM T60631 C8NBS0 135242318 IC50 = 44 nM T60631 CZ7J9V 135497783 IC50 = 1000 nM T60631 C3IJ9V 135497787 IC50 = 1000 nM T60631 CK0RB4 135497790 IC50 = 2990 nM T60631 C9YNE7 135497791 IC50 = 1000 nM T60631 C8HO5W 135497794 IC50 > 10000 nM T60631 CSP15M 135497800 IC50 > 100000 nM T60631 C0S3KJ 135497814 IC50 > 10000 nM T60631 C3J8WZ 135497817 IC50 = 111 nM T60631 CJ3FI8 135497818 IC50 = 410 nM T60631 C6LJ4F 135497822 IC50 = 375 nM T60631 C2U8QZ 135497823 IC50 = 190 nM T60631 CERT86 135497824 IC50 = 475 nM T60631 C2HAP4 135497831 IC50 = 100000 nM T60631 CBF73U 135497834 IC50 > 100000 nM T60631 C1FA6Q 135497835 IC50 = 201 nM T60631 C2D0BL 135497840 IC50 = 218 nM T60631 CEKY53 135497841 IC50 = 1000 nM T60631 CH34CP 135497843 IC50 = 36 nM T60631 CW8MO3 135497844 IC50 = 38 nM T60631 C7GKS9 135497849 IC50 = 106 nM T60631 C3WKV4 135497850 IC50 = 390 nM T60631 CU8T6K 135497853 IC50 > 100000 nM T60631 CC58VR 135497854 IC50 > 10000 nM T60631 C0ML5X 135497855 IC50 = 1000 nM T60631 C1PJB2 135497865 IC50 > 100000 nM T60631 C1V9AZ 135497869 IC50 = 410 nM T60631 CN2W4U 135497870 IC50 = 1230 nM T60631 C03CVQ 135497872 IC50 = 1227 nM T60631 C03EJP 135497876 IC50 = 1000 nM T60631 CR09SN 135497877 IC50 > 100000 nM T60631 CU6T8C 135497878 IC50 > 100000 nM T60631 C45KEI 135497879 IC50 = 1100 nM T60631 CWFT86 135497881 IC50 = 150 nM T60631 CB8G6M 135497884 IC50 = 1268 nM T60631 CK5G2W 135510524 IC50 = 140 nM T60631 CR51FT 135511450 IC50 = 63800 nM T60631 CI47VJ 135566923 IC50 = 20 nM T60631 CHA4N2 136013680 IC50 > 10 nM T60631 C7O9XA 136026002 IC50 = 10000 nM T60631 C61JVA 136026154 IC50 = 1073 nM T60631 CIJ3Q6 136068594 IC50 = 104 nM T60631 CK09OF 136086925 IC50 = 1000 nM T60631 C2G9XA 136086927 IC50 = 100000 nM T60631 C1Y0PS 136118031 IC50 > 100000 nM T60631 CA76XZ 136118032 IC50 > 100000 nM T60631 CVQ41X 136118033 IC50 > 100000 nM T60631 CU5XR2 136118034 IC50 > 100000 nM T60631 C4G6PT 136118035 IC50 = 3230 nM T60631 CDT7E4 136211077 IC50 > 100 nM T60631 C1YUD0 136219394 IC50 > 10 nM T60631 CIU8W3 136254389 IC50 > 10 nM T60631 C5OSN2 137148836 IC50 = 3680 nM T60631 CXC69T 137321158 IC50 = 66 nM T60631 C25ERN 137631967 IC50 = 0.04 nM T60631 CGRF93 137632798 IC50 = 416 nM T60631 CB43LI 137633642 IC50 = 236 nM T60631 CA41YB 137633865 IC50 = 2695 nM T60631 CI1E8V 137634241 IC50 = 379 nM T60631 C6W9JQ 137634508 IC50 = 162 nM T60631 C5SY7W 137636232 IC50 = 62.5 nM T60631 C06JRX 137637094 IC50 = 0.2 nM T60631 C9C8QW 137641230 IC50 = 4803 nM T60631 C7TG3J 137641313 IC50 = 616.6 nM T60631 C1AC7S 137642462 IC50 = 3395 nM T60631 C87DGP 137644408 IC50 = 410 nM T60631 C2H9FD 137644986 IC50 = 102 nM T60631 CCV0K4 137648368 IC50 = 631 nM T60631 C41BJA 137649417 IC50 = 2224 nM T60631 CA2J1F 137649865 IC50 = 1661 nM T60631 C1DK0P 137651391 IC50 = 0.4 nM T60631 C28QUP 137652864 IC50 = 89.5 nM T60631 COVM63 137652906 IC50 = 139 nM T60631 CQ63RS 137654616 IC50 = 61.2 nM T60631 CRQX04 137654763 IC50 = 78 nM T60631 CLW48N 137656611 IC50 = 1639 nM T60631 CV5H3Z 137657932 IC50 = 0.7 nM T60631 CPV1S9 137658287 IC50 = 387 nM T60631 CR4IV1 137660865 IC50 = 1259 nM T60631 C4H3JQ 137662071 IC50 = 104 nM T60631 C6AK0N 139030518 IC50 = 34 nM T60631 C29XUO 145945978 IC50 > 1000 nM T60631 C4HB8M 145949394 IC50 = 152 nM T60631 C0V8SM 145954139 IC50 = 7.6 nM T60631 CS2NR4 145964261 IC50 = 2.8 nM T60631 C65YWX 145964882 IC50 = 440 nM T60631 CHC3T0 145965031 IC50 > 10000 nM T60631 CP92ZF 145965329 IC50 = 50 nM T60631 C9Y7DO 145965819 IC50 = 20.7 nM T60631 C9HXI4 145966620 IC50 = 600 nM T60631 CQE9M5 145966810 IC50 = 60 nM T60631 C1EH6C 145967078 IC50 = 1200 nM T60631 C4OD9Q 145967187 IC50 = 20.3 nM T60631 CDW83M 145967332 IC50 = 162.8 nM T60631 CWJ12M 145969155 IC50 = 6 nM T60631 CGW5S1 145969844 IC50 = 900 nM T60631 CB8R3A 145970271 IC50 > 10000 nM T60631 COJ7H5 145970527 IC50 = 0.2 nM T60631 CNDL79 145970990 IC50 = 0.4 nM T60631 CJD5Q1 145972024 IC50 = 0.7 nM T60631 CO5Z4B 145972302 IC50 = 22.2 nM T60631 C40VIL 145972979 IC50 = 160 nM T60631 CQBY19 145974023 IC50 = 6200 nM T60631 CF59KI 145976265 IC50 = 0.6 nM T60631 CZB63Y 145976371 IC50 = 0.7 nM T60631 C4X7CT 145977420 IC50 = 4000 nM T60631 CLA57T 145978300 IC50 = 430 nM T60631 C1RTZ4 145983560 IC50 = 32500 nM T60631 C9WA3P 145983862 IC50 = 6070 nM T60631 CBRK57 145985435 IC50 = 19000 nM T60631 CB74GU 145985813 IC50 = 5510 nM T60631 C03PYD 145986466 IC50 < 1000 nM T60631 CK56ME 145994823 IC50 = 51 nM T60631 CE4FH2 146018674 IC50 = 19 nM T60631 CP9W6A 154729143 IC50 = 20 nM T60631 CUZ9R5 155510459 IC50 = 880 nM T60631 C2MD1Q 155513187 IC50 > 10000 nM T60631 CXN58S 155521337 IC50 = 29000 nM T60631 C1RA6C 155524092 IC50 = 1600 nM T60631 CI15ZX 155526266 IC50 = 350 nM T60631 C45BJK 155526700 IC50 = 1100 nM T60631 C8I6SB 155529587 IC50 = 7600 nM T60631 CS69CA 155532132 IC50 = 5.2 nM T60631 CKE7Y9 155533164 IC50 = 44 nM T60631 CM0U3I 155534552 IC50 > 1000 nM T60631 CGZJ65 155538203 IC50 = 660 nM T60631 CSJ01Q 155538965 IC50 = 300 nM T60631 C2KR0V 155545994 IC50 = 1500 nM T60631 C5DV7N 155546585 IC50 = 200 nM T60631 CIR16L 155548076 IC50 = 63000 nM T60631 C3MQW4 155548639 IC50 = 360 nM T60631 CAR40G 155551366 IC50 = 1140 nM T60631 C84JMI 155552727 IC50 = 6700 nM T60631 COS2F3 155569572 IC50 = 560 nM T60631 D00ATA 5908088 IC50 = 460 nM T60631 D02BXJ 46864270 IC50 = 0.2 nM T60631 D02NNT 53232451 IC50 = 19 nM T60631 D03BQI 3794 IC50 = 720 nM T60631 D03DZO 11715767 IC50 > 10000 nM T60631 D03EHM 24905142 IC50 < 1 nM T60631 D06HVH 54613583 IC50 = 7700 nM T60631 D07OSK 6419834 IC50 = 760 nM T60631 D08HFG 24809764 IC50 > 10000 nM T60631 D09HVH 135566652 IC50 > 10 nM T60631 D0A1CM 5281855 IC50 > 40000 nM T60631 D0CE3R 5312137 IC50 = 770 nM T60631 D0E7VO 59627005 IC50 < 100 nM T60631 D0H1OK 11562302 Ki = 407 nM T60631 D0HE0E 5941540 IC50 = 1100 nM T60631 D0KH5T 5687 IC50 = 4.5 nM T60631 D0L3FK 5289419 IC50 = 1600 nM T60631 D0M4QA 56935577 IC50 = 1.3 nM T60631 D0N4LR 53469448 IC50 = 1215 nM T60631 D0Q0YV 24944925 IC50 = 11481.54 nM T60631 D0Q4EQ 16742063 IC50 = 183 nM T60631 D0R2WK 16038120 EC50 > 1000 nM T60631 D0T8NU 16757525 IC50 > 4000 nM T60631 D0U3NI 53246941 IC50 = 161 nM T60631 D0US9O 45275255 IC50 = 46 nM T60631 D0W4UQ 46233144 IC50 = 5300 nM T60631 D0Y1UL 10561847 IC50 = 2300 nM T58266 D0E3TC 44259 IC50 = 137 nM T58266 C7YG1N 24759534 IC50 = 21 nM T58266 CE1A9V 57394653 IC50 = 434 nM T58266 CXJ63M 59603829 IC50 = 29 nM T58266 CQEU96 59603842 IC50 = 2.9 nM T58266 CV63UL 67240318 IC50 > 10000 nM T58266 C5DGR9 69036886 IC50 = 10000 nM T58266 C1HW4B 89735655 IC50 = 16000 nM T58266 C9WGB8 127035904 IC50 = 3100 nM T58266 CXC69T 137321158 IC50 = 233 nM T58266 C2MD1Q 155513187 IC50 > 10000 nM T58266 D05FXD 44478401 IC50 = 4.5 nM T58266 D0X8BU 71718651 IC50 = 1500 nM T61400 D00HGB 4488 IC50 = 17000 nM T61400 D08ROP 3899 IC50 = 10000 nM T61400 D09SOA 28718 IC50 = 13000 nM T61400 D00LSI 9820008 IC50 = 134 nM T61400 D0G7UX 5284373 IC50 > 50000 nM T61400 D0N3XT 57030 IC50 = 6 nM T61400 CYIU47 1543 IC50 = 7 nM T61400 CI9TK0 3884 IC50 = 100 nM T61400 CR6HO1 8593 IC50 = 144000 nM T61400 CU4O3D 38081 IC50 = 8000 nM T61400 C5LA7B 76864 IC50 = 709 nM T61400 CE2KN9 130331 Ki = 25 nM T61400 CYRV23 131419 IC50 = 12 nM T61400 CS74HZ 145726 IC50 = 12380 nM T61400 C4U5MD 202918 IC50 = 10000 nM T61400 C21UMY 271388 IC50 = 541 nM T61400 CT6MA7 322307 IC50 > 10000 nM T61400 CP4ZX0 459316 IC50 = 420 nM T61400 CVY91W 517728 IC50 > 100000 nM T61400 CEVD28 517858 IC50 > 100000 nM T61400 C9JAF2 523003 IC50 > 200000 nM T61400 CO0MN5 609454 IC50 > 20000 nM T61400 CZH54C 615334 IC50 > 20000 nM T61400 C14CXW 619026 IC50 = 3960 nM T61400 CJ1W4Q 623973 IC50 = 3410 nM T61400 COPS41 653193 IC50 > 100000 nM T61400 CDX0O4 660996 IC50 > 200000 nM T61400 CXS49M 669445 IC50 = 6830 nM T61400 CZO9S8 673239 IC50 = 13010 nM T61400 C4UOR0 673730 IC50 = 5176.8 nM T61400 CCLM40 684865 IC50 = 930 nM T61400 CG2Q8Y 736801 IC50 = 18280 nM T61400 C5UJV1 739902 IC50 = 1830 nM T61400 C8S6ZO 741601 IC50 > 100000 nM T61400 C23WHO 741604 IC50 > 100000 nM T61400 C76COZ 743061 IC50 > 200000 nM T61400 CFD56M 753240 IC50 = 1566.1 nM T61400 CE6G1W 777184 IC50 > 100000 nM T61400 CS4BA6 777191 IC50 > 100000 nM T61400 CFD0U2 780529 IC50 = 17750 nM T61400 C4GAY3 813108 IC50 = 15620 nM T61400 C2PSU0 831397 IC50 = 780 nM T61400 CC4S8F 844231 IC50 = 550 nM T61400 CC0MD2 865225 Ki > 500 nM T61400 CIQ10J 904019 IC50 = 3249.8 nM T61400 CH52WR 947453 IC50 = 9074 nM T61400 CBT92O 993994 IC50 = 136.2 nM T61400 CSBU38 1027581 IC50 = 1270 nM T61400 C9JCR6 1037067 IC50 = 340 nM T61400 CQYE56 1133093 IC50 = 5900 nM T61400 C3O5MX 1223586 IC50 = 57.1 nM T61400 C87PLH 1223597 IC50 = 666.2 nM T61400 C8HS9K 1374134 IC50 = 1130 nM T61400 COV67N 1432578 IC50 = 400 nM T61400 CG1F9T 1460771 IC50 > 100000 nM T61400 CM4L5I 1481799 IC50 = 17400 nM T61400 C1KT8C 1746237 IC50 = 260 nM T61400 CR3IN2 1746284 IC50 = 1310 nM T61400 CGDC52 1763612 IC50 = 436.7 nM T61400 C5S6NK 1830299 IC50 = 250 nM T61400 CYA5F2 1965647 IC50 = 89000 nM T61400 C8NMY3 2063288 IC50 = 51 nM T61400 C93GMJ 2578400 IC50 > 20000 nM T61400 C9HOI8 2709135 IC50 = 12400 nM T61400 C31KAP 2743369 IC50 = 39000 nM T61400 C7GE9J 2759386 IC50 = 1040 nM T61400 CH25IU 2858282 IC50 > 10000 nM T61400 CS0KO4 2995335 IC50 = 16080 nM T61400 CN0MT1 3100461 IC50 = 29 nM T61400 CX2L9S 3227262 IC50 > 100000 nM T61400 CS7MF9 3851642 Ki = 17900 nM T61400 C54XIU 3899945 IC50 = 1600 nM T61400 C01OYK 4221076 Ki = 35900 nM T61400 CR9A1Q 4605417 IC50 > 500000 nM T61400 C8JYO2 4749758 IC50 = 3848 nM T61400 CMSE21 5057449 IC50 = 9.7 nM T61400 C1TC3N 5167181 Ki = 28 nM T61400 CJ1BM6 5184531 IC50 > 200000 nM T61400 CU73XG 5287459 Ki = 2800 nM T61400 CK86XL 5308416 IC50 > 100000 nM T61400 CYP02U 5376552 IC50 = 10000 nM T61400 CM4A3N 7346373 IC50 = 81 nM T61400 CNY5I0 7416167 IC50 > 100000 nM T61400 CE5XO9 7688340 IC50 = 1300 nM T61400 C67CZW 7955004 IC50 = 1358 nM T61400 C9KT2N 8850862 IC50 > 100000 nM T61400 C0LYE6 9045495 IC50 > 20000 nM T61400 C0KG4F 9173919 IC50 > 10000 nM T61400 CCGE73 9547914 IC50 = 280 nM T61400 CQ70AU 9824035 Ki = 4 nM T61400 CHZ34C 9861992 IC50 = 303 nM T61400 C0XCI6 9948506 IC50 = 410 nM T61400 CNP6S9 10000399 Ki = 13 nM T61400 CG7EM6 10029745 Ki = 26 nM T61400 CRA6E7 10048413 Ki = 4 nM T61400 CA7TO9 10064328 IC50 = 700 nM T61400 C1EF4U 10342449 IC50 = 33 nM T61400 CB4D0C 10356750 IC50 > 100000 nM T61400 CJ1KH3 10364016 Ki = 8.4 nM T61400 C3S6CZ 10404208 IC50 = 800 nM T61400 CIO0Z9 10454174 IC50 = 8 nM T61400 CZ4KA1 10457096 IC50 = 7 nM T61400 C68KRG 10488180 IC50 > 50000 nM T61400 C5ZE1V 10491179 IC50 = 3600 nM T61400 CI31FC 10492984 IC50 > 50000 nM T61400 C4N5YT 10494611 IC50 = 6060 nM T61400 CCFG07 10496492 IC50 > 50000 nM T61400 C6REV7 10512886 IC50 = 19400 nM T61400 COVK03 10515945 IC50 > 50000 nM T61400 CC1K4I 10516844 IC50 > 50000 nM T61400 CM15VH 10516983 IC50 = 500 nM T61400 CU5PT2 10519719 IC50 > 50000 nM T61400 C54GLO 10540764 IC50 = 6200 nM T61400 C54IJE 10541884 IC50 = 6500 nM T61400 C0PLE3 10544308 IC50 > 50000 nM T61400 C32DIH 10565707 IC50 = 4000 nM T61400 CED3A9 10565785 IC50 > 50000 nM T61400 CY1RS4 10587807 IC50 > 50000 nM T61400 CLXD24 10587934 IC50 > 50000 nM T61400 C42WEO 10635802 IC50 = 2700 nM T61400 CHDR60 10643787 Ki = 6000 nM T61400 C81RJI 10657722 IC50 = 16500 nM T61400 CZ4DH9 10680043 IC50 = 12100 nM T61400 C6ZNV5 10680597 IC50 = 3200 nM T61400 C4X0UR 10682218 IC50 = 22400 nM T61400 CQ96TA 10687946 Ki = 3700 nM T61400 CH1UQ6 10690749 Ki = 4000 nM T61400 C15GIF 10691466 Ki > 100000000 nM T61400 CI5AT8 10703799 IC50 > 50000 nM T61400 C21DPI 10710291 IC50 > 50000 nM T61400 C1H3PI 10711746 IC50 > 50000 nM T61400 CZQH50 10738106 Ki > 100000000 nM T61400 CIG1Q0 10752727 IC50 = 9000 nM T61400 CJ1ED3 10755169 IC50 > 50000 nM T61400 C27DHQ 10759123 IC50 > 50000 nM T61400 CU26LB 10759927 IC50 > 50000 nM T61400 CU29BN 10800984 IC50 = 22500 nM T61400 CX5EL6 10805428 IC50 > 50000 nM T61400 C6O0EX 10808375 IC50 = 239 nM T61400 CIW5B8 10825617 IC50 = 2600 nM T61400 CUZ3X1 10828593 IC50 > 50000 nM T61400 C3HM9N 10829333 IC50 > 50000 nM T61400 CDV5Q8 10830186 IC50 > 50000 nM T61400 CRZH97 10830342 Ki = 4000 nM T61400 CY53LI 10849345 IC50 > 50000 nM T61400 CBRS89 10852951 Ki = 20000 nM T61400 C3PU1H 10853437 IC50 = 784 nM T61400 C4VCG7 10895558 Ki = 32 nM T61400 CRJ4Q5 10929378 Ki = 331 nM T61400 C2Q8UR 10938858 Ki = 12 nM T61400 CV1KX4 11016730 Ki = 8 nM T61400 CL4CV9 11038663 Ki = 1500 nM T61400 C87CWY 11102808 Ki = 6 nM T61400 CVGQ92 11135071 Ki = 2400 nM T61400 CMW42X 11416123 Ki = 203 nM T61400 C1D5CH 11524688 IC50 = 1 nM T61400 C5IEU6 11530041 IC50 > 200000 nM T61400 C4C1QF 11703683 IC50 > 200000 nM T61400 CKS30M 11762691 Ki = 138 nM T61400 C6NY3W 11825758 Ki = 91 nM T61400 CUB8Y3 12454047 Ki = 15100 nM T61400 CE6Z4B 13960629 Ki = 60 nM T61400 COMT87 13960632 Ki = 29 nM T61400 CK5RC6 13960639 Ki = 30 nM T61400 C51BST 13960640 Ki = 20 nM T61400 C2GNU0 13960650 Ki = 10 nM T61400 C0UX8F 13960654 Ki = 13 nM T61400 CYJ08U 13960663 Ki = 220 nM T61400 C4XWV8 13960668 Ki = 10 nM T61400 C0QF9I 13960681 Ki = 270 nM T61400 C7T2LK 14222046 IC50 = 2800 nM T61400 CJQS85 14498146 IC50 = 5 nM T61400 CP17YT 14498150 IC50 = 10 nM T61400 CZ9B2W 14498162 IC50 = 312 nM T61400 CZ13DK 14498163 IC50 = 211 nM T61400 CU29XS 14498165 IC50 = 217 nM T61400 CXB50A 14498174 IC50 = 6 nM T61400 CW3P1R 14498175 IC50 = 7 nM T61400 CR7KX9 14498179 IC50 = 18 nM T61400 C1ORM4 14773532 Ki = 17 nM T61400 CL3M4G 15858807 IC50 > 50000 nM T61400 CQN40R 15942657 IC50 = 44 nM T61400 CP2WJ3 15942658 IC50 = 2 nM T61400 CXV7A5 16099894 IC50 = 306000 nM T61400 COH7N2 16099900 IC50 = 151000 nM T61400 C8D0KF 16099905 IC50 = 72000 nM T61400 CM8CL1 16099913 IC50 = 56000 nM T61400 C3UK7A 16099914 IC50 = 136000 nM T61400 C3V2KY 16099916 IC50 = 212000 nM T61400 CR5EY8 16099917 IC50 = 17000 nM T61400 CBE84I 16099918 IC50 = 51000 nM T61400 C31XCS 16099919 IC50 = 283000 nM T61400 C2FXW0 16099923 IC50 = 26000 nM T61400 CFY05L 16099926 IC50 = 230000 nM T61400 CO5SY7 16099929 IC50 = 4000 nM T61400 COSK93 16099935 IC50 = 135000 nM T61400 C51NZE 16099968 IC50 = 301000 nM T61400 C2NH3G 16099971 IC50 = 41000 nM T61400 C0IBF1 16099978 IC50 = 32000 nM T61400 C8HGF0 16100002 IC50 = 134000 nM T61400 CUM26S 16100003 IC50 = 141000 nM T61400 C4ZVE0 16100004 IC50 = 130000 nM T61400 CUMK61 16100005 IC50 = 270 nM T61400 CDG5U9 16100006 IC50 = 132000 nM T61400 CE39KU 16100011 IC50 = 43000 nM T61400 C7VE4W 16100015 IC50 = 4900 nM T61400 CJM54Z 16102641 Ki = 3630 nM T61400 CZX30A 16102642 Ki = 60400 nM T61400 CKT91D 16102643 IC50 > 500000 nM T61400 CMEU86 16102644 Ki = 27 nM T61400 COQW13 16102645 Ki = 12800 nM T61400 CL3A8Z 16102646 IC50 > 500000 nM T61400 CXO5U1 16210733 IC50 = 1440 nM T61400 CXUO14 16457485 IC50 = 46000 nM T61400 C83SPM 16457486 IC50 = 12000 nM T61400 C8MSK3 16777509 IC50 > 200000 nM T61400 CD20AH 21084669 IC50 = 42 nM T61400 CA9Z7Y 21084690 IC50 = 225 nM T61400 CI1T5W 21084721 IC50 = 170 nM T61400 C37ANI 21084723 IC50 = 45 nM T61400 CDS2T7 21084730 IC50 = 110 nM T61400 C1XP7M 21084734 IC50 = 90 nM T61400 CL46XF 21084739 IC50 = 310 nM T61400 C06TFS 21084741 IC50 = 11 nM T61400 C6XJ2K 21084746 IC50 = 8400 nM T61400 C58MIH 21084752 IC50 = 17 nM T61400 CI41ZH 21084760 IC50 = 1700 nM T61400 CHE52U 21084763 IC50 = 5700 nM T61400 C0B6YR 21084801 IC50 = 127 nM T61400 CK7N2M 21084803 IC50 = 2000 nM T61400 C1AW4H 21084857 IC50 = 105 nM T61400 CND19K 21084860 IC50 = 173 nM T61400 C38QSO 21084861 IC50 = 667 nM T61400 C6QYE9 22042531 IC50 = 680 nM T61400 C8RBW0 22042533 IC50 = 1460 nM T61400 CP09OF 22431257 IC50 > 100000 nM T61400 CK02UJ 22433941 IC50 > 100000 nM T61400 C0I8AV 22577320 IC50 > 100000 nM T61400 C09MTF 22579221 IC50 > 100000 nM T61400 C5AR8O 23647298 Ki > 100000000 nM T61400 CS0RU6 23647299 IC50 = 3 nM T61400 CZAT30 23647300 IC50 = 9 nM T61400 C29UME 23647301 IC50 = 12 nM T61400 C8Y6DJ 23647302 IC50 = 1000 nM T61400 CWFG85 23647303 IC50 = 10 nM T61400 C6GOR3 23647305 IC50 > 1000 nM T61400 CUJ9D8 23647306 IC50 > 1000 nM T61400 CQOP01 23647307 IC50 > 1000 nM T61400 C8GJ7K 23647308 IC50 = 16 nM T61400 C9AVR7 23647309 IC50 = 340 nM T61400 C3WMP9 23663733 Ki = 24 nM T61400 CG5YM6 23663964 Ki = 12 nM T61400 C7KBU5 23668107 Ki = 15 nM T61400 CQYE41 23668976 Ki = 8.3 nM T61400 CK7MW5 23671800 Ki = 40 nM T61400 CT3AJ5 23671801 Ki = 17 nM T61400 CN3FK4 23673359 Ki = 8 nM T61400 CP01FB 23673369 Ki = 38 nM T61400 CE9OD6 23673384 Ki = 24 nM T61400 CRK25G 23673385 Ki = 210 nM T61400 CR59ZP 23673428 Ki = 230 nM T61400 CT7XA2 23686481 Ki = 170 nM T61400 CB94XJ 23693316 Ki = 31 nM T61400 C1HEK3 23699178 Ki = 4.5 nM T61400 C5T0GQ 23699179 Ki > 130 nM T61400 C96KCH 23699180 Ki = 27 nM T61400 CR2KJ1 23699181 Ki = 26 nM T61400 CL3ZU5 23699195 Ki = 25 nM T61400 C2E0MI 23699196 Ki = 52 nM T61400 CWE6Z3 24829334 IC50 = 2.999 nM T61400 CJ3Z9A 24882111 IC50 > 200000 nM T61400 CZVG60 24882112 IC50 > 200000 nM T61400 CD26YW 24882113 IC50 > 200000 nM T61400 C4WDG1 24882114 IC50 > 200000 nM T61400 C5T0WI 24882115 IC50 > 200000 nM T61400 CO39XG 24882194 IC50 > 200000 nM T61400 C8RBY3 24882195 IC50 > 200000 nM T61400 CMW12Z 24882196 IC50 > 200000 nM T61400 C5YZR8 24882197 IC50 > 200000 nM T61400 C5QHJ4 24882198 IC50 > 200000 nM T61400 CYV89J 24986460 IC50 = 87.9 nM T61400 CUN1P0 24986824 IC50 = 15 nM T61400 C38QGT 24986825 IC50 = 19.01 nM T61400 C8WCI6 24986827 IC50 = 89.95 nM T61400 C5JQG2 24987180 IC50 = 149.97 nM T61400 C35LNQ 24987183 IC50 = 19.01 nM T61400 CJ03WL 24987187 IC50 = 14 nM T61400 CS62EF 24987532 IC50 = 199.99 nM T61400 CS4BW8 24987910 IC50 = 11.99 nM T61400 CP1R6W 24987911 IC50 = 99.08 nM T61400 CDR80K 24987915 IC50 = 109.9 nM T61400 CXB25G 24987916 IC50 = 11.99 nM T61400 CGZU50 24988290 IC50 = 32.96 nM T61400 CTG18W 24988292 IC50 = 5.998 nM T61400 CM2L0X 24988658 IC50 = 5 nM T61400 CG75AI 24988659 IC50 = 17.02 nM T61400 CD35ZG 24988663 IC50 = 52.97 nM T61400 CDEO28 24988664 IC50 = 23.01 nM T61400 C92RNP 24989025 IC50 = 3.999 nM T61400 CE3L9I 24989026 IC50 = 7.998 nM T61400 C06BXV 24989027 IC50 = 10.99 nM T61400 CN5ZM2 24989028 IC50 = 3.999 nM T61400 CY7L9T 24989029 IC50 = 5.998 nM T61400 CIY92Z 24989389 IC50 = 5 nM T61400 CHAV93 24991946 IC50 = 199.99 nM T61400 CDH5W8 25263414 IC50 > 100000 nM T61400 CB15SF 25263431 IC50 > 100000 nM T61400 CL3SD8 25263432 IC50 > 100000 nM T61400 C5Z3US 25263434 IC50 > 100000 nM T61400 COLC28 25495325 IC50 = 1987 nM T61400 CWZ9H4 25706226 IC50 = 500 nM T61400 C8R0MH 32617117 IC50 > 100000 nM T61400 CPG2Q9 33839737 IC50 > 20000 nM T61400 CZ4XT5 33839743 IC50 > 20000 nM T61400 CQW1K4 39168487 IC50 = 139 nM T61400 C7F3ZH 44131574 IC50 > 100000 nM T61400 C5VN0T 44131575 IC50 > 100000 nM T61400 CUAJ90 44131922 IC50 > 100000 nM T61400 CM7AW1 44133588 IC50 > 100000 nM T61400 C5K7IB 44133769 IC50 > 100000 nM T61400 CN2TB0 44133775 IC50 > 100000 nM T61400 CKB5I7 44133952 IC50 > 100000 nM T61400 CI9K2W 44133953 IC50 > 100000 nM T61400 CR1CK8 44133954 IC50 > 100000 nM T61400 C7Y1KS 44285497 Ki = 48 nM T61400 CY6S8F 44285498 Ki = 420 nM T61400 CBP4T6 44285510 Ki = 500 nM T61400 CK65QM 44285511 Ki > 500 nM T61400 CZ8FV0 44285515 Ki = 150 nM T61400 CWF16G 44285691 Ki > 500 nM T61400 CN9G7I 44285758 Ki = 210 nM T61400 CZ9SR1 44285816 Ki > 500 nM T61400 C4CS3W 44285821 Ki = 140 nM T61400 C4OKR6 44285831 Ki = 63 nM T61400 CQ1YE7 44285854 Ki > 500 nM T61400 C29KGA 44285869 Ki > 500 nM T61400 CMSA39 44285877 Ki > 500 nM T61400 C2GRM9 44285885 Ki > 500 nM T61400 CJN7W1 44285921 Ki > 500 nM T61400 CCJF78 44285965 Ki = 1.7 nM T61400 CP2K8U 44286040 Ki > 500 nM T61400 CX29PC 44286041 Ki > 500 nM T61400 C35FSI 44286043 Ki > 500 nM T61400 CVAQ16 44286046 Ki > 500 nM T61400 C0CW6B 44286047 Ki = 400 nM T61400 CFU27H 44286048 Ki = 210 nM T61400 C49DIP 44286071 Ki > 500 nM T61400 CK0U7D 44286092 Ki > 500 nM T61400 C9PHU1 44286125 Ki = 40 nM T61400 C8Y3PW 44286140 Ki = 300 nM T61400 C12MXQ 44286187 Ki = 390 nM T61400 C6JR5L 44286221 Ki = 50 nM T61400 C1GB4Q 44286358 Ki > 500 nM T61400 C2ZNO0 44286361 Ki = 200 nM T61400 C4KNW7 44286387 Ki = 56 nM T61400 CQ6EO9 44293728 Ki > 1000 nM T61400 C3B8RJ 44293730 Ki > 430 nM T61400 CPI71Q 44293941 Ki = 21 nM T61400 C1QN8U 44293943 Ki > 200 nM T61400 C5D7ME 44293959 Ki = 83 nM T61400 CCT29I 44293961 Ki = 34 nM T61400 CS83WH 44293976 Ki > 1000 nM T61400 C8O4XR 44294171 Ki = 22 nM T61400 CHW1N3 44294190 Ki = 240 nM T61400 C8RP4O 44294214 Ki > 390 nM T61400 CT43AI 44294217 Ki = 30 nM T61400 C7IQE3 44294221 Ki = 71 nM T61400 CPB80C 44294227 Ki = 24 nM T61400 C5CHG6 44294237 Ki = 330 nM T61400 C7KX3C 44294295 Ki > 200 nM T61400 CX1UO6 44294412 Ki = 23 nM T61400 C0R2CT 44294414 Ki = 32 nM T61400 C0KBU1 44294426 Ki = 40 nM T61400 CZR59L 44294460 Ki = 30 nM T61400 C0I6AW 44294461 Ki = 25 nM T61400 CA8CK0 44310310 IC50 = 3200 nM T61400 CQN0O6 44310311 IC50 = 40400 nM T61400 CN0W2Z 44310325 IC50 = 11000 nM T61400 CKX9M2 44310351 IC50 > 50000 nM T61400 C8VU2D 44310352 IC50 > 50000 nM T61400 C82UGB 44310357 IC50 = 35000 nM T61400 C42QUC 44310364 IC50 > 50000 nM T61400 C1NDM3 44310365 IC50 > 50000 nM T61400 C8NYB2 44310373 IC50 = 7200 nM T61400 C8L9GJ 44310374 IC50 = 3000 nM T61400 CFR1N4 44310375 IC50 > 50000 nM T61400 CW2P0E 44310381 IC50 > 50000 nM T61400 C97IWD 44310382 IC50 > 50000 nM T61400 CB09NP 44310384 IC50 > 50000 nM T61400 CJI6L4 44310624 IC50 > 50000 nM T61400 CQ80RE 44310640 IC50 = 9300 nM T61400 C2BV7J 44310695 IC50 > 50000 nM T61400 CSV6U2 44310717 IC50 > 50000 nM T61400 CSKY53 44310718 IC50 > 50000 nM T61400 CZPH40 44310719 IC50 > 50000 nM T61400 CPC91U 44310720 IC50 > 50000 nM T61400 CQ63ML 44336155 Ki = 25 nM T61400 CKJG53 44336188 Ki = 81 nM T61400 CON4J0 44336227 Ki = 380 nM T61400 CJ36QM 44336238 Ki = 160 nM T61400 CV2YP1 44336240 Ki = 10 nM T61400 CBR56T 44336242 Ki = 40 nM T61400 CCOD06 44336252 Ki = 34 nM T61400 C6MDQ8 44336254 Ki = 13 nM T61400 CTNU65 44336258 Ki = 27 nM T61400 CXN9R0 44336260 Ki > 182 nM T61400 C53DQP 44336262 Ki = 20 nM T61400 C4XTY9 44336266 Ki = 206 nM T61400 CE9WV6 44336282 Ki = 139 nM T61400 CYU8D2 44336303 Ki > 1000 nM T61400 CJ4IO9 44336305 Ki = 962 nM T61400 CB04QY 44336310 Ki = 218 nM T61400 CU1J9K 44336317 Ki = 300 nM T61400 CI64RV 44336322 Ki > 204 nM T61400 CTG26W 44336326 Ki = 370 nM T61400 C3LW2N 44336350 Ki = 190 nM T61400 C7W0GM 44336357 Ki = 409 nM T61400 CZP09Q 44336370 Ki > 180 nM T61400 CFN50P 44336420 Ki = 55 nM T61400 C72IQU 44336436 Ki = 59 nM T61400 CQX43F 44336438 Ki = 43 nM T61400 C1TR0G 44336445 Ki = 135 nM T61400 CHG3Z0 44336456 Ki = 37 nM T61400 CH6C5E 44336469 Ki = 48 nM T61400 C0K4EJ 44369486 IC50 = 50 nM T61400 CZL2G9 44369512 IC50 = 70 nM T61400 C6ZVK8 44369554 IC50 = 610 nM T61400 CD96TQ 44369555 IC50 = 370 nM T61400 C4CNL3 44369573 IC50 = 18 nM T61400 C5OZC9 44369738 IC50 = 290 nM T61400 C1QY9G 44369747 IC50 = 150 nM T61400 CD0S8A 44369748 IC50 = 20 nM T61400 CF05RS 44369749 IC50 = 610 nM T61400 CE9D2I 44369777 IC50 = 2900 nM T61400 C0RMF9 44369833 IC50 = 390 nM T61400 CWM3B8 44369844 IC50 = 735 nM T61400 CLA7T9 44369868 IC50 = 180 nM T61400 C05AET 44369870 IC50 = 80 nM T61400 CGI86U 44369871 IC50 = 840 nM T61400 CUM5Y3 44403188 IC50 = 41 nM T61400 CM43HR 44403223 IC50 = 3800 nM T61400 C9QEN3 44403229 IC50 = 360 nM T61400 CGUB91 44403235 IC50 = 131 nM T61400 CH2I7M 44403236 IC50 = 11 nM T61400 CW0BM2 44403240 IC50 = 205 nM T61400 CY6L2E 44403243 IC50 = 15 nM T61400 CCEQ67 44403250 IC50 = 58 nM T61400 CGJQ91 44403251 IC50 = 4 nM T61400 C23ZOD 44406354 IC50 = 10 nM T61400 CIDY35 44409277 Ki > 100000000 nM T61400 CA1PQ7 44480861 IC50 > 30000 nM T61400 C1TPI7 44541920 IC50 = 19000 nM T61400 C3SOX5 44542366 IC50 = 28000 nM T61400 C6SX0K 44631844 IC50 = 100 nM T61400 C3R9WV 44631846 IC50 = 5500 nM T61400 CAM34R 45484114 IC50 = 9800 nM T61400 C4HL9F 46200812 IC50 = 1.5 nM T61400 C9H2VC 46352384 IC50 > 100000 nM T61400 CP32ID 46945388 IC50 = 750 nM T61400 CH1BZ9 51031042 IC50 = 2100 nM T61400 CX20SO 51347101 IC50 > 100000 nM T61400 C2DB3K 51347103 IC50 > 100000 nM T61400 C7LA9W 51347104 IC50 > 30000 nM T61400 C7D0BN 51347106 IC50 > 100000 nM T61400 C8Y2TG 51347246 IC50 > 50000 nM T61400 CXYM16 51347247 IC50 > 50000 nM T61400 C2LBF4 51347391 IC50 > 50000 nM T61400 CLD8K7 51347393 IC50 > 100000 nM T61400 CSNY98 51347394 IC50 > 100000 nM T61400 CA3Y7Q 51347395 IC50 > 100000 nM T61400 CBL8I4 51347396 IC50 > 100000 nM T61400 CD3A8K 51347397 IC50 > 100000 nM T61400 C50NBU 51347540 IC50 > 100000 nM T61400 CN6GR1 51347541 IC50 > 100000 nM T61400 CR0P6T 51347542 IC50 > 100000 nM T61400 CGZ1A8 51347543 IC50 > 100000 nM T61400 C8TM7G 51347544 IC50 = 17000 nM T61400 CET37V 51347545 IC50 = 2100 nM T61400 C6B5MK 51347546 IC50 > 100000 nM T61400 C14BCJ 51347692 IC50 > 100000 nM T61400 CX75YQ 51347695 IC50 > 100000 nM T61400 CB1YV6 51347852 IC50 > 50000 nM T61400 CS6NB1 51349275 IC50 = 41000 nM T61400 C1MC4Y 51349276 IC50 = 7000 nM T61400 CU8GP0 53257300 IC50 > 100000 nM T61400 C0TL1W 53259245 IC50 > 100000 nM T61400 C0VR6N 53357599 IC50 = 36 nM T61400 C7T2YD 53362039 IC50 = 103 nM T61400 CX3Z8F 53392537 IC50 > 100000 nM T61400 CWN60M 53392616 IC50 > 100000 nM T61400 CZ64LI 53392617 IC50 > 100000 nM T61400 C48LJO 53392618 IC50 > 100000 nM T61400 C3EYX4 53392619 IC50 > 100000 nM T61400 C1BI6K 53392620 IC50 > 100000 nM T61400 C07IOL 53392704 IC50 > 100000 nM T61400 C2VRT7 53392705 IC50 > 100000 nM T61400 CW21EC 53392883 IC50 > 100000 nM T61400 C8CHL6 53392884 IC50 > 100000 nM T61400 CI2A8R 54585315 IC50 > 100000 nM T61400 CIDY47 54650356 IC50 > 50000 nM T61400 CX9D6Z 54684419 Ki = 14 nM T61400 C0D2XW 54714524 IC50 = 200 nM T61400 CU5LE1 54727973 Ki = 22 nM T61400 C7NCJ6 54727974 Ki = 21 nM T61400 CT7SP0 54727975 Ki = 25 nM T61400 C7PS2J 54727976 Ki = 40 nM T61400 C1SBV6 54727977 Ki = 2000 nM T61400 C2C6YU 54727978 Ki = 190 nM T61400 CPE81B 54727979 Ki = 10700 nM T61400 C4IPZ2 54727980 Ki = 2.7 nM T61400 C4P2EB 54727981 Ki = 23 nM T61400 C9RIT4 54727982 Ki = 25 nM T61400 C97HOU 54727983 Ki = 16 nM T61400 CIKS61 54727984 Ki = 39 nM T61400 C3AJ2O 54727985 Ki = 16 nM T61400 CZK51H 57328384 IC50 = 1300 nM T61400 C0ZF1L 57328385 IC50 = 200 nM T61400 C2Z0ND 57393100 IC50 > 9900 nM T61400 C62JOU 57396592 IC50 > 9900 nM T61400 CI25UB 57396593 IC50 > 9900 nM T61400 C58IAE 57398368 IC50 = 5700 nM T61400 CWQI09 57398380 IC50 > 9900 nM T61400 CZAG81 57400035 IC50 = 1100 nM T61400 C3MB2N 57401837 IC50 = 6300 nM T61400 CJZ62H 57403545 IC50 > 9900 nM T61400 C5W7RH 57825994 IC50 > 100000 nM T61400 C3VPE9 58284833 IC50 > 30000 nM T61400 CBF5P4 58284844 IC50 > 30000 nM T61400 CBNY54 58284845 IC50 > 30000 nM T61400 CB6WD8 58284852 IC50 > 30000 nM T61400 C1FG6A 58284878 IC50 > 30000 nM T61400 C2TK4P 58284891 IC50 > 30000 nM T61400 C6QK1F 58284898 IC50 = 15100 nM T61400 C9VR6E 58284899 IC50 > 30000 nM T61400 CQ43AI 58284908 IC50 > 30000 nM T61400 CH7JY4 58284909 IC50 > 30000 nM T61400 C7WVD5 60143791 IC50 = 7900 nM T61400 CK8EN9 60166357 IC50 = 29000 nM T61400 CFRP36 60166358 IC50 = 32000 nM T61400 C14ACE 60166481 IC50 = 63000 nM T61400 CHI8V5 60166482 IC50 = 9500 nM T61400 CG68AW 60166483 IC50 = 6500 nM T61400 CNP12G 60166484 IC50 = 18000 nM T61400 C5SVK6 60166485 IC50 = 51 nM T61400 CZ6K2Y 60166486 IC50 = 30000 nM T61400 CZJ3V1 60166487 IC50 = 13000 nM T61400 CZA1F7 60166617 IC50 = 13 nM T61400 CA2LX1 60166618 IC50 > 100000 nM T61400 CPZ1N5 60166619 IC50 > 100000 nM T61400 C1S4FV 60166620 IC50 > 100000 nM T61400 CLK3E2 70681098 IC50 = 7300 nM T61400 C52JHL 70681099 IC50 = 14900 nM T61400 CZB37T 70681849 IC50 = 6800 nM T61400 CE40MY 70685307 IC50 > 30000 nM T61400 CWIC42 70685308 IC50 > 30000 nM T61400 C64XSH 70685311 IC50 = 3100 nM T61400 CJ03MS 70685312 IC50 > 30000 nM T61400 CSX35W 70687453 IC50 = 5600 nM T61400 CL98PO 70689508 IC50 = 17200 nM T61400 CZ24SU 71457078 IC50 > 100000 nM T61400 CKP71J 71460750 IC50 > 100000 nM T61400 CD8S7U 71543403 IC50 = 18 nM T61400 CU28IZ 71768298 IC50 > 20000 nM T61400 CQW30K 71768301 IC50 = 7400 nM T61400 CS58YD 71768302 IC50 = 910 nM T61400 C3KTN1 71768303 IC50 > 20000 nM T61400 CKE08I 71768304 IC50 = 560 nM T61400 C6H5MU 71768305 IC50 > 20000 nM T61400 CK2GQ1 71768306 IC50 = 3600 nM T61400 CYKP52 71768307 IC50 = 1500 nM T61400 CZ7U6C 71768308 IC50 = 9500 nM T61400 C1U9BT 71768309 IC50 = 1900 nM T61400 CT3BZ6 71768310 IC50 = 2700 nM T61400 CJ4N6E 71768311 IC50 > 20000 nM T61400 CFQU69 71768313 IC50 = 8900 nM T61400 CV8NP3 71812412 IC50 = 10000 nM T61400 CI38XK 71816353 IC50 = 1 nM T61400 C6YT1I 71816637 IC50 = 19 nM T61400 C5UHP7 71816638 IC50 = 16 nM T61400 C3JT2L 71817130 IC50 = 310 nM T61400 CQH7D2 71817131 IC50 = 95 nM T61400 CZE85V 73291708 IC50 = 2600 nM T61400 C8GOQ7 85469100 IC50 >= 200000 nM T61400 C0Y5AD 90644862 IC50 = 940 nM T61400 CR4FW7 90644863 IC50 = 1090 nM T61400 CPXR78 90644864 IC50 = 1500 nM T61400 CQ42AS 90644865 IC50 = 3210 nM T61400 C6FWV8 90644866 IC50 = 3440 nM T61400 C5T1CM 90644867 IC50 = 4580 nM T61400 CS83LW 90644868 IC50 = 6090 nM T61400 CB3E6M 90644869 IC50 = 2280 nM T61400 CJSX56 90644870 IC50 = 2830 nM T61400 CAQ06B 90665760 IC50 > 200000 nM T61400 CP85ZC 90665761 IC50 > 200000 nM T61400 CY2V9O 90665762 IC50 > 200000 nM T61400 C4MUT5 90665763 IC50 > 200000 nM T61400 CZR4C7 90665764 IC50 > 200000 nM T61400 C8CL1E 90665765 IC50 > 200000 nM T61400 CB2ES5 90665766 IC50 > 200000 nM T61400 C3G2UO 90665767 IC50 = 130000 nM T61400 CJLC28 90665769 IC50 > 200000 nM T61400 CIE5D9 90665770 IC50 > 200000 nM T61400 CZHP65 90665771 IC50 > 200000 nM T61400 C14DXE 90665772 IC50 > 200000 nM T61400 CTPM46 90665774 IC50 > 200000 nM T61400 CTNB32 90665775 IC50 > 200000 nM T61400 CBX34M 90665776 IC50 > 200000 nM T61400 CN21UQ 90665777 IC50 > 200000 nM T61400 CSB93Z 91885568 IC50 > 100000 nM T61400 C2HD7Z 91995955 IC50 = 35 nM T61400 CWL6G0 100253413 IC50 = 969 nM T61400 C5COZ3 101593774 IC50 = 911 nM T61400 C61WAN 118096600 IC50 = 58 nM T61400 CGU37E 118096604 IC50 = 26 nM T61400 CZKA39 118430456 IC50 = 25 nM T61400 C4YLQ5 118430504 IC50 = 12.59 nM T61400 CTZ40W 118430507 IC50 = 15.85 nM T61400 CHQ6T4 118430570 IC50 = 0.7943 nM T61400 CJT5K7 118430627 IC50 = 125.89 nM T61400 CUYJ02 118732492 IC50 = 3649 nM T61400 CD4H3U 118732493 IC50 = 2346 nM T61400 CVJF50 118732494 IC50 = 1926 nM T61400 CJ1P9X 118732495 IC50 = 562 nM T61400 CKJZ07 118732496 IC50 > 10000 nM T61400 CM4ED7 118732497 IC50 = 887 nM T61400 CC6UJ1 118732498 IC50 = 2111 nM T61400 C69UCS 118732499 IC50 > 10000 nM T61400 CSX9V2 118732500 IC50 > 10000 nM T61400 CQW9A3 118732501 IC50 = 6040 nM T61400 CUT04K 118732502 IC50 = 9028 nM T61400 C2BN7S 118732503 IC50 > 10000 nM T61400 CA7LO0 118732504 IC50 = 325 nM T61400 CC76FZ 118732505 IC50 = 645 nM T61400 CVB0D1 118732506 IC50 = 372 nM T61400 CK4L0N 118732507 IC50 = 515 nM T61400 CGJ32E 118732508 IC50 = 652 nM T61400 C60EIK 118732509 IC50 = 552 nM T61400 CTV35M 118732510 IC50 = 49 nM T61400 C4UOA8 118732511 IC50 = 408 nM T61400 CJK3H2 118732512 IC50 = 284 nM T61400 CZFP14 118732513 IC50 = 131 nM T61400 CF30NS 118732514 IC50 = 128 nM T61400 CALH84 118732515 IC50 = 174 nM T61400 CCR2H0 118732516 IC50 = 393 nM T61400 C7TQ3K 118732517 IC50 > 10000 nM T61400 CA02BG 118732518 IC50 = 1108 nM T61400 CB6M0L 118732519 IC50 = 453 nM T61400 CK3P5B 118732520 IC50 > 10000 nM T61400 C6Q5VR 118732521 IC50 > 10000 nM T61400 C2YTD6 118732522 IC50 > 10000 nM T61400 C20RZO 118732523 IC50 > 10000 nM T61400 CK90CH 118732524 IC50 = 311 nM T61400 CQG43L 118732525 IC50 > 10000 nM T61400 CTR2E0 118732526 IC50 > 10000 nM T61400 C5UQ2W 118732527 IC50 > 10000 nM T61400 CL5FB9 121232409 IC50 > 10000 nM T61400 CM0D9K 121596187 IC50 > 50000 nM T61400 CYEG40 122182176 IC50 = 210 nM T61400 CPZL16 122182177 IC50 = 1380 nM T61400 C4S9IA 122182178 IC50 = 32000 nM T61400 CC5R3U 122182179 IC50 = 300 nM T61400 CEFS97 122182180 IC50 = 28 nM T61400 C8XLA4 122182181 IC50 = 13 nM T61400 CLMP60 122182182 IC50 = 47000 nM T61400 CT7W5H 122182183 IC50 = 7800 nM T61400 CX2N6P 122182187 IC50 = 20000 nM T61400 C0CIL6 122182188 IC50 = 28000 nM T61400 CQN24Y 122182309 IC50 = 50000 nM T61400 CAT68V 122182311 IC50 = 37000 nM T61400 C3TGE0 122182312 IC50 = 51000 nM T61400 C25RGB 122182313 IC50 = 42000 nM T61400 CMS2L7 122182314 IC50 = 56000 nM T61400 CKS81I 122182315 IC50 = 20000 nM T61400 C4I7SQ 122182317 IC50 = 40000 nM T61400 C90HTM 122182318 IC50 = 55000 nM T61400 CFG4A1 122182320 IC50 = 31000 nM T61400 C78KCO 122182321 IC50 = 48000 nM T61400 CG2TM5 122182323 IC50 = 38000 nM T61400 CRW8H4 122182324 IC50 = 23000 nM T61400 CE19LW 122552662 IC50 > 100000 nM T61400 C53HXW 124219453 IC50 = 2680 nM T61400 CO5MJ2 124220265 IC50 = 45 nM T61400 CPE3W5 129012054 IC50 > 10000 nM T61400 C7BZ2C 129892319 IC50 = 29 nM T61400 CB4L7A 132157886 IC50 = 28 nM T61400 C8MCQ4 132157904 IC50 = 14 nM T61400 CL20KI 132157920 IC50 = 8 nM T61400 C2DHO4 132157940 IC50 = 59 nM T61400 C4VSN2 132157947 IC50 = 11 nM T61400 CQ3B8W 132157950 IC50 = 8 nM T61400 CE6R2J 132157951 IC50 = 2 nM T61400 C1XN0P 132157952 IC50 = 66 nM T61400 CE28UI 132157962 IC50 = 93 nM T61400 CN60JA 132157967 IC50 = 87 nM T61400 CCMB41 132157980 IC50 = 24 nM T61400 CU43LK 132157983 IC50 = 19 nM T61400 CN3G5T 132157984 IC50 = 15 nM T61400 C7VWA6 132158000 IC50 = 9 nM T61400 CCP58M 132158011 IC50 = 425 nM T61400 CCUD94 132158017 IC50 = 356 nM T61400 C0TEG4 133107894 IC50 = 26.2 nM T61400 C6I5PQ 133107895 IC50 = 28.3 nM T61400 CEDN72 134131421 IC50 = 1060 nM T61400 CWT12E 134132121 IC50 = 472 nM T61400 C8M1QP 134132231 IC50 > 5000 nM T61400 CYCP47 134132411 IC50 = 293 nM T61400 CK5Y4P 134132509 IC50 = 2400 nM T61400 C3K8ZH 134132554 IC50 = 638 nM T61400 CJ42KU 134132701 IC50 > 625 nM T61400 C0OS1M 134132798 IC50 = 2570 nM T61400 C5VHD9 134132876 IC50 = 2600 nM T61400 C3U7FP 134133701 IC50 = 764 nM T61400 C7N8TB 134133820 IC50 > 1250 nM T61400 C65APX 134134172 IC50 = 284 nM T61400 C30OTN 134134345 IC50 = 719 nM T61400 CL7J1T 134134663 IC50 = 68.1 nM T61400 C7MRI8 134134984 IC50 = 5.77 nM T61400 CB46GN 134135152 IC50 = 44.3 nM T61400 C8PCZ2 134135269 IC50 = 147 nM T61400 CXM5V0 134136454 IC50 > 625 nM T61400 CHJY85 134136646 IC50 = 16.8 nM T61400 CYT6F0 134137084 IC50 = 1785 nM T61400 CY6M8K 134137428 IC50 > 1250 nM T61400 C9YBH7 134138544 IC50 = 434 nM T61400 CA1I7E 134138701 IC50 = 44.3 nM T61400 CWRE28 134139256 IC50 = 496 nM T61400 CH3NZ2 134139862 IC50 > 1000 nM T61400 CF46NK 134140808 IC50 = 11.4 nM T61400 C6AC9N 134140885 IC50 = 46.2 nM T61400 CW70VS 134141087 IC50 > 5000 nM T61400 C6S5RU 134141210 IC50 > 1000 nM T61400 CABX80 134141331 IC50 = 40.4 nM T61400 CKD2N9 134141516 IC50 = 839 nM T61400 CFR2J0 134141914 IC50 > 5000 nM T61400 C1IEJ4 134142176 IC50 > 1000 nM T61400 C73QKY 134142713 IC50 = 277 nM T61400 CYMD98 134142784 IC50 > 5000 nM T61400 C7X5OI 134143212 IC50 = 20.6 nM T61400 C8RAT6 134143381 IC50 = 2510 nM T61400 CB8O2I 134143841 IC50 = 23.9 nM T61400 CW3Q8P 134143855 IC50 = 434 nM T61400 CVX30C 134144166 IC50 = 204 nM T61400 C5XAR8 134144586 IC50 > 625 nM T61400 C8GJL6 134145423 IC50 = 47.8 nM T61400 CH2I3N 134146144 IC50 > 250 nM T61400 C1VBL4 134146300 IC50 = 524 nM T61400 CYXB69 134146530 IC50 = 16.6 nM T61400 C6E0XS 134146866 IC50 > 1000 nM T61400 CME12V 134146963 IC50 = 297 nM T61400 CM1YL6 134147611 IC50 = 2222 nM T61400 CC3WM4 134148792 IC50 = 31.5 nM T61400 C57TUY 134148877 IC50 = 2790 nM T61400 C16HPS 134148955 IC50 > 5000 nM T61400 C6ELV9 134149204 IC50 = 52.1 nM T61400 C4D6LF 134149443 IC50 = 39.8 nM T61400 C2X8SQ 134149497 IC50 = 2070 nM T61400 C6D2QA 134150022 IC50 > 1000 nM T61400 CR7U1Q 134150360 IC50 = 22.5 nM T61400 CBL3R7 134150906 IC50 = 4.14 nM T61400 CID91E 134151822 IC50 = 968 nM T61400 CM50OK 134151915 IC50 = 1274 nM T61400 C24AXS 134151955 IC50 = 389 nM T61400 CSFV61 134152327 IC50 > 5000 nM T61400 CV6D4L 134152813 IC50 = 13.3 nM T61400 C5J1RB 134152933 IC50 > 500 nM T61400 C10LBV 134153435 IC50 = 3960 nM T61400 CF14TP 134153573 IC50 = 20.3 nM T61400 CVG3B9 134154001 IC50 > 1250 nM T61400 CZ7LC8 134154436 IC50 = 0.97 nM T61400 CZP9N7 134154785 IC50 = 77.5 nM T61400 CN45AT 134155043 IC50 > 5000 nM T61400 CH0G8V 134155982 IC50 > 625 nM T61400 COV89K 134156366 IC50 = 82.4 nM T61400 C6I3BD 134156999 IC50 > 5000 nM T61400 CCE1I9 134157042 IC50 = 152 nM T61400 CKE10V 134157478 IC50 = 46.1 nM T61400 C6QU0R 134157954 IC50 = 1972 nM T61400 C43SAY 134686803 IC50 = 1.2 nM T61400 C4D6EY 135393504 IC50 > 200000 nM T61400 CY5HF3 135449276 IC50 > 50000 nM T61400 C2KYZ4 135547547 IC50 = 6 nM T61400 CPIK81 135547548 IC50 = 2100 nM T61400 CC76EY 135547549 IC50 = 7 nM T61400 CCR5D0 136094765 IC50 = 676 nM T61400 C2NP1R 136094766 IC50 = 178 nM T61400 C1RD6K 136109168 Ki = 11 nM T61400 CDY3F5 137228155 IC50 = 4850 nM T61400 C50MRK 137641335 IC50 > 100000 nM T61400 CY6P4D 137653786 IC50 > 100000 nM T61400 C2SN9G 144675334 IC50 > 10000 nM T61400 CWG3H6 144675341 IC50 > 10000 nM T61400 CXU86F 144675343 IC50 = 4410 nM T61400 C6Y5JR 144675358 IC50 = 8510 nM T61400 C2E6HP 145953041 IC50 > 5000 nM T61400 C4YWQ5 145954585 IC50 = 480 nM T61400 C3V6AM 145954937 IC50 = 43 nM T61400 C6HS3D 145955655 IC50 = 4.3 nM T61400 CR9S7T 145967579 IC50 = 36 nM T61400 CRD48N 145967592 IC50 = 8400 nM T61400 CP5T7R 145967609 IC50 = 504 nM T61400 C2L8ER 145967629 IC50 = 54.3 nM T61400 C9YXD8 145967714 IC50 = 2790 nM T61400 CP53CF 145967883 IC50 > 50000 nM T61400 CJ92MV 145967884 IC50 > 200000 nM T61400 C6AWO9 145967932 IC50 = 259 nM T61400 CBE08Q 145968095 IC50 = 7550 nM T61400 CIO84W 145968108 IC50 = 22.1 nM T61400 CK3AV2 145968283 IC50 = 32.7 nM T61400 C7HR3S 145968438 IC50 = 9.71 nM T61400 CG07KW 145968498 IC50 = 12500 nM T61400 CSWU25 145968738 IC50 = 165 nM T61400 CTX53Y 145968746 IC50 = 54.2 nM T61400 CI4M6R 145968875 IC50 = 11.8 nM T61400 CKP9F3 145969000 IC50 = 10100 nM T61400 CC48ZB 145969067 IC50 = 21.2 nM T61400 CP83ZU 145969133 IC50 > 200000 nM T61400 C1CRY2 145969257 IC50 > 200000 nM T61400 CQJN68 145969266 IC50 = 184 nM T61400 CH04GY 145969286 IC50 = 5260 nM T61400 C46BMT 145969345 IC50 = 165 nM T61400 C3US4M 145969551 IC50 = 74.4 nM T61400 C1OA6H 145969566 IC50 = 1220 nM T61400 CB6UJ0 145969586 IC50 > 200000 nM T61400 CEF9G4 145969676 IC50 = 1420 nM T61400 CTO5L0 145969709 IC50 = 2480 nM T61400 CRD6A0 145969747 IC50 = 373 nM T61400 CCSW79 145969925 IC50 = 391 nM T61400 C91JZX 145969991 IC50 = 1430 nM T61400 CC0FJ1 145970351 IC50 = 235 nM T61400 C5K1TO 145970373 IC50 = 8070 nM T61400 CE51XM 145970439 IC50 > 200000 nM T61400 CBR39P 145970472 IC50 = 201 nM T61400 CF1D6A 145970592 IC50 = 3310 nM T61400 CBZ7K2 145970897 IC50 = 8210 nM T61400 C1UP2Z 145970932 IC50 > 200000 nM T61400 C04OZP 145971128 IC50 = 148 nM T61400 CE5WF0 145971993 IC50 = 35 nM T61400 CFNA78 145973351 IC50 = 760 nM T61400 CKJ05B 145978954 IC50 = 10640 nM T61400 C42DTN 145979421 IC50 > 10000 nM T61400 CM63NF 145979727 IC50 > 10000 nM T61400 C6CD7V 145979986 IC50 > 10000 nM T61400 CMJN90 145980028 IC50 > 10000 nM T61400 CN8L1H 145981260 IC50 = 3030 nM T61400 C8QAE1 145981477 IC50 > 10000 nM T61400 CR2X6E 145981868 IC50 > 10000 nM T61400 CQ4V3U 145982007 IC50 > 10000 nM T61400 CRTG43 145986592 IC50 = 127 nM T61400 CXBW37 145986714 IC50 > 10000 nM T61400 C7US0K 145987016 IC50 > 10000 nM T61400 C0O3PH 145987908 IC50 > 10000 nM T61400 C62CRS 145988488 IC50 > 10000 nM T61400 C0QPI7 145988677 IC50 = 1750 nM T61400 CMA7F1 145989710 IC50 = 79.4 nM T61400 C4DRW5 145991341 IC50 = 1120 nM T61400 C4LR1H 145991562 IC50 > 10000 nM T61400 CZRE38 145992417 IC50 > 10000 nM T61400 C64JTQ 145993462 IC50 = 9450 nM T61400 CBQ2W1 145993607 IC50 > 10000 nM T61400 C70RLZ 145994006 IC50 > 10000 nM T61400 CQ31LZ 146672982 IC50 = 330 nM T61400 CL7C6B 155511813 IC50 > 200000 nM T61400 C64RXS 155512621 IC50 = 7480 nM T61400 CVNP52 155522278 IC50 > 250000 nM T61400 CAMY59 155522616 IC50 = 808 nM T61400 C10DUW 155525976 IC50 > 250000 nM T61400 CHAZ73 155526511 IC50 = 2100 nM T61400 C4GM2N 155528177 IC50 = 15480 nM T61400 CPG08O 155528245 IC50 = 1560 nM T61400 CX6MI9 155530572 IC50 > 200000 nM T61400 C2GBC6 155530731 IC50 = 1960 nM T61400 C5RAT1 155535476 IC50 = 108 nM T61400 CIN03T 155536717 IC50 = 4600 nM T61400 C4VBM7 155538807 IC50 = 3600 nM T61400 C4FAQ0 155539488 IC50 > 250000 nM T61400 CT57BM 155539527 IC50 > 250000 nM T61400 CVG89J 155542108 IC50 = 41000 nM T61400 C1EJR7 155543412 IC50 = 1220 nM T61400 CGH72R 155550183 IC50 >= 200000 nM T61400 C1Q6JR 155550675 IC50 = 123 nM T61400 CRI9P6 155552167 IC50 = 1050 nM T61400 C81JEO 155552732 IC50 = 13440 nM T61400 C1FNG7 155553026 IC50 = 3700 nM T61400 CVY7T5 155565603 IC50 = 3340 nM T61400 C2BQF8 155566700 IC50 = 7370 nM T61400 C9KER8 155567039 IC50 = 1800 nM T61400 D00YPH 10239 IC50 = 12000 nM T61400 D01NWQ 823850 Ki = 50900 nM T61400 D03QKF 44631845 IC50 = 700 nM T61400 D04HZA 23647297 Ki = 1100 nM T61400 D05SXU 13707619 Ki = 1800 nM T61400 D06IPT 54727972 Ki = 11 nM T61400 D0C1NU 799096 Ki = 64400 nM T61400 D0HQ1I 777193 IC50 > 200000 nM T61400 D0M2EM 4650 IC50 = 34000 nM T61400 D0R1GF 914489 Ki = 700 nM T61400 D0V1EK 735838 IC50 > 10000 nM T32369 D07HBX 338 EC50 > 250000 nM T32369 D0TQ1G 5071 IC50 = 11000 nM T32369 C2HNF8 8369 IC50 > 199526.23 nM T32369 CBIR94 10313 IC50 > 500000 nM T32369 C1E6AF 10665 IC50 > 500000 nM T32369 CO1VU5 68129 IC50 = 22500 nM T32369 CPFG50 69521 IC50 = 17100 nM T32369 C2TXC4 69732 IC50 > 500000 nM T32369 C5UI8E 72871 EC50 > 250000 nM T32369 C21QXO 97273 IC50 = 800000 nM T32369 C6QHP0 129682 IC50 = 4700 nM T32369 CBZ21G 231363 EC50 > 250000 nM T32369 COV46I 412786 IC50 > 500000 nM T32369 C84QRW 493418 IC50 = 5400 nM T32369 CRTA37 514101 IC50 = 100000 nM T32369 CWM5V2 514102 IC50 = 710000 nM T32369 C17NCI 514103 IC50 > 500000 nM T32369 CN2QU6 514104 IC50 > 500000 nM T32369 C7Q1NU 514105 IC50 > 1000000 nM T32369 CT70CJ 514106 IC50 = 9000 nM T32369 CJS2H4 514107 IC50 = 8000 nM T32369 CM1F9C 514108 IC50 = 29000 nM T32369 C68EOP 514109 IC50 = 11000 nM T32369 C9Q5GX 514111 IC50 = 17000 nM T32369 CQN35A 514114 IC50 = 45000 nM T32369 C7M3LZ 514115 IC50 = 10000 nM T32369 C4FET6 514116 IC50 = 48000 nM T32369 C4A3FL 514117 IC50 = 50000 nM T32369 C70GSU 514118 IC50 = 40000 nM T32369 C3H9AU 514119 IC50 = 9500 nM T32369 CS59VC 514120 IC50 = 20000 nM T32369 C2XKU8 514121 IC50 = 38000 nM T32369 C2I7QU 514122 IC50 = 3000 nM T32369 CX8LN4 514123 IC50 = 40000 nM T32369 CVN46B 514124 IC50 = 50000 nM T32369 CRB09A 514125 IC50 = 10000 nM T32369 CU0GV9 514126 IC50 = 10000 nM T32369 CIPK34 514129 IC50 = 18000 nM T32369 CW82IF 514130 IC50 = 35000 nM T32369 CC1M3U 516699 IC50 > 500000 nM T32369 C1TL8Y 676116 EC50 > 250000 nM T32369 C61EIH 720992 IC50 = 63000 nM T32369 CTN40Q 3010943 IC50 = 19700 nM T32369 CIQ9G2 3642111 IC50 = 9700 nM T32369 C3T7EQ 5271788 Ki = 960 nM T32369 C6KOC4 5278545 IC50 = 85000 nM T32369 C7RG3L 5496307 Ki = 480 nM T32369 COF29Y 6479289 IC50 = 29400 nM T32369 C5DY7C 6479290 IC50 > 500000 nM T32369 CH5NM6 6479291 Ki = 90 nM T32369 C4NKV9 6479293 IC50 = 26000 nM T32369 CX12FK 6479294 IC50 = 9500 nM T32369 CVSY49 6479295 IC50 = 8000 nM T32369 C2ZN5V 6508940 IC50 = 307000 nM T32369 CI1EZ6 9794049 IC50 = 95000 nM T32369 C0OE3C 10397916 IC50 = 18000 nM T32369 CR1WA9 10511097 IC50 > 50000 nM T32369 CYK0W1 10883256 IC50 = 38000 nM T32369 C0AF6P 10959579 IC50 = 14000 nM T32369 CJ3T2W 11565002 IC50 = 3981.07 nM T32369 C3KSA4 11644313 IC50 = 2700 nM T32369 CE5N1C 11822161 Ki = 280 nM T32369 CPAX91 12280547 IC50 = 3981.07 nM T32369 CPTF25 14668277 IC50 = 32000 nM T32369 CB73ST 16072595 IC50 = 940 nM T32369 CDSJ73 19009433 IC50 = 12589.25 nM T32369 C2Q9MB 20463660 IC50 = 3162.28 nM T32369 COW47N 21661241 IC50 = 4800 nM T32369 CID6E7 40637838 EC50 > 250000 nM T32369 CQ0HV4 44591820 IC50 = 31622.78 nM T32369 CRQY52 53326350 IC50 = 1500 nM T32369 C3J8QS 54736410 IC50 = 588 nM T32369 CG1UO2 56945147 IC50 = 47.8 nM T32369 CLCR86 58067149 IC50 = 241 nM T32369 CRV36F 58067162 IC50 = 164 nM T32369 CZPF90 60152398 IC50 = 17800 nM T32369 CV7TF4 67471511 IC50 = 419 nM T32369 C2K3NO 67471576 IC50 = 115 nM T32369 C17QSM 67471579 IC50 = 103 nM T32369 C9I2UH 67471599 IC50 = 116 nM T32369 CZF5C7 67471604 IC50 = 110 nM T32369 CA6L5Z 67471613 IC50 = 239 nM T32369 CQB7Y5 67471799 IC50 = 281 nM T32369 C2PF7J 68096633 IC50 = 80.4 nM T32369 CLB73C 68096640 IC50 = 358 nM T32369 CZAT10 68096717 IC50 = 286 nM T32369 CG30DK 68097098 IC50 = 114 nM T32369 CPK0U5 70681844 IC50 > 200000 nM T32369 CNR02U 70681845 IC50 > 200000 nM T32369 CN6U2E 70683948 IC50 > 200000 nM T32369 CA7N0C 70683949 IC50 > 200000 nM T32369 CL9VM5 70683950 IC50 > 200000 nM T32369 C34JGW 70686071 IC50 > 200000 nM T32369 CBV81D 70686072 IC50 > 200000 nM T32369 CXI3P9 70686073 IC50 > 200000 nM T32369 CQJZ59 70686074 IC50 > 200000 nM T32369 C6XNH2 70686075 IC50 > 200000 nM T32369 CX45TL 70688763 IC50 = 600 nM T32369 CM4QR3 70688764 IC50 = 2100 nM T32369 C4CT7U 70690222 IC50 > 200000 nM T32369 CCR6H3 70690223 IC50 > 200000 nM T32369 CJ03XD 70690224 IC50 > 200000 nM T32369 C9UFV4 70690225 IC50 > 200000 nM T32369 C5CT3X 70692391 IC50 > 200000 nM T32369 C80AEI 70692392 IC50 > 200000 nM T32369 CAIY09 70692393 IC50 > 200000 nM T32369 CSQ87I 70692394 IC50 > 200000 nM T32369 CHS6R4 70692395 IC50 > 200000 nM T32369 C0FIQ3 70692985 IC50 = 31 nM T32369 CX36GS 70692986 IC50 = 100 nM T32369 CHJ0L7 70694446 IC50 > 200000 nM T32369 CT9LM8 70696513 IC50 > 200000 nM T32369 CC2O6Y 70696514 IC50 > 200000 nM T32369 CD46SX 71685911 IC50 = 5011.87 nM T32369 CDS41B 86725691 IC50 = 1584.89 nM T32369 CF6LB5 89475995 IC50 = 460 nM T32369 C94SIP 90429399 IC50 = 5 nM T32369 C2TIB0 90672508 IC50 = 7943.28 nM T32369 CC81GD 90672509 IC50 = 3981.07 nM T32369 CVM7C5 90924450 IC50 = 68600 nM T32369 C7BVQ9 91900676 IC50 = 12 nM T32369 CDFE74 123130720 IC50 = 2500 nM T32369 CGU63O 129115717 IC50 = 4800 nM T32369 C9OLI2 130014282 IC50 = 3981.07 nM T32369 CFE5P7 130407610 IC50 = 19952.62 nM T32369 C5GLQ2 130407621 IC50 = 12589.25 nM T32369 C3Z0ER 130407634 IC50 = 2900 nM T32369 CGD4X9 130407636 IC50 = 12589.25 nM T32369 CZ1R5L 130407637 IC50 = 6300 nM T32369 C1GIW9 130407660 IC50 > 50000 nM T32369 C2JNL8 130407758 IC50 = 2511.89 nM T32369 CRO2J9 130407768 IC50 = 320 nM T32369 C51NLR 130407789 IC50 = 730 nM T32369 CJ3HW7 130407797 IC50 > 50000 nM T32369 CU45HA 130407803 IC50 > 100000 nM T32369 COD41A 130407819 IC50 = 940 nM T32369 C5TQ9S 130407824 IC50 = 14 nM T32369 C24VAX 130407831 IC50 = 794.33 nM T32369 C4Q2RB 130407849 IC50 < 50118.72 nM T32369 CF90GR 130407852 IC50 = 2200 nM T32369 CMUC01 130407853 IC50 = 610 nM T32369 CWRX97 130407858 IC50 = 3900 nM T32369 C7WBV6 130407859 IC50 = 1000 nM T32369 C7ULM2 130407876 IC50 = 1500 nM T32369 CM2D3C 130407878 IC50 = 1995.26 nM T32369 CM0LH3 130407896 IC50 = 3162.28 nM T32369 C7A1SO 130407903 IC50 = 1800 nM T32369 CDIS43 130407905 IC50 > 50000 nM T32369 CBJD59 130407909 IC50 = 12589.25 nM T32369 C1B7YA 130407915 IC50 = 360 nM T32369 C5RB9A 130407917 IC50 = 3400 nM T32369 CI9S4Q 130407921 IC50 = 120 nM T32369 C7KBY3 130407941 IC50 = 10000 nM T32369 CX6D8T 130407957 IC50 = 3162.28 nM T32369 CTA2O9 130407971 IC50 = 36 nM T32369 C4QS8K 130407983 IC50 = 180 nM T32369 C5PZY1 130407996 IC50 = 190 nM T32369 C0TMF8 130408003 IC50 = 1995.26 nM T32369 CNM91W 130408004 IC50 = 5011.87 nM T32369 CLN1U2 130410573 IC50 = 1350 nM T32369 CSM78J 130423169 IC50 = 5011.87 nM T32369 CBEC68 130423208 IC50 = 3800 nM T32369 C0CS7X 130423209 IC50 = 4.8 nM T32369 CD7XK5 130423213 IC50 = 2.3 nM T32369 CNO27Z 130423214 IC50 < 1.995 nM T32369 CK61PJ 130423218 IC50 < 1.995 nM T32369 C8Z5KB 130423922 IC50 = 15.85 nM T32369 C7JO8Y 130423987 IC50 = 5.012 nM T32369 C87WPY 130424055 IC50 = 501.19 nM T32369 CEOQ59 130424056 IC50 = 398.11 nM T32369 CID81V 130424057 IC50 = 125.89 nM T32369 CHR9G6 130424060 IC50 = 398.11 nM T32369 C5IJP6 130424161 IC50 = 1258.93 nM T32369 CZ60AB 130424162 IC50 = 1000 nM T32369 C1IMB8 130424164 IC50 = 2300 nM T32369 C7GHV8 130424166 IC50 = 5011.87 nM T32369 CJO72A 130424167 IC50 = 794.33 nM T32369 CBN43F 130424170 IC50 > 100000 nM T32369 C2HES8 130424264 IC50 = 25 nM T32369 C2SMJ4 135427888 Ki = 1100 nM T32369 C8N4DY 135446125 Ki = 8000 nM T32369 CVSF86 135446253 Ki = 50420 nM T32369 CBP8L3 135446970 Ki = 1840 nM T32369 CJL7F5 135566706 Ki = 5010 nM T32369 CVWM42 135566707 Ki = 18700 nM T32369 CKC68W 135566866 IC50 = 11 nM T32369 C6Q8UW 135691141 IC50 = 8300 nM T32369 C1PJ2Y 135788271 Ki = 49000 nM T32369 C9AHX0 136244213 Ki = 20300 nM T32369 CWK6Q3 136244214 Ki = 3556 nM T32369 C98VRQ 136244215 Ki = 11200 nM T32369 CJF6E5 136244216 Ki = 24300 nM T32369 COIZ90 136244267 Ki = 990 nM T32369 CW23BY 136244268 Ki = 720 nM T32369 C4ZV9G 136244269 Ki = 1000 nM T32369 C3NS6L 136254246 Ki = 7100 nM T32369 CU07AY 136254247 Ki = 1200 nM T32369 C9T0WA 136254248 EC50 > 250000 nM T32369 C2BYO6 136254249 Ki = 2280 nM T32369 C56VXI 136254250 Ki = 290 nM T32369 CI4CY8 136254251 Ki = 1610 nM T32369 CVX61S 136254252 Ki = 1392 nM T32369 CPEH10 136254253 Ki = 21600 nM T32369 C2B8SH 136254254 Ki = 38600 nM T32369 C1XBR9 136254255 Ki = 28570 nM T32369 CE8V2B 136254256 Ki = 70500 nM T32369 CAU12K 136254257 Ki = 1650 nM T32369 C7SU8O 136254258 EC50 > 250000 nM T32369 C30YVF 137215899 IC50 < 2 nM T32369 C6R9PF 138455151 IC50 < 2 nM T32369 CS28UI 138455152 IC50 < 1.995 nM T32369 CB3RM4 138455153 IC50 = 0.1259 nM T32369 C0P6OS 138539091 IC50 = 6 nM T32369 C79SMD 138539163 IC50 = 0.1 nM T32369 C4U1DS 138539180 IC50 = 2.3 nM T32369 C84WET 138539264 IC50 = 3.162 nM T32369 CBQ3D8 138539265 IC50 < 1.995 nM T32369 CE85SC 138539266 IC50 = 0.2512 nM T32369 C3AK1B 138539267 IC50 = 3.162 nM T32369 CA8UE5 138539270 IC50 = 12.59 nM T32369 C6Q9BN 138539273 IC50 = 6.3 nM T32369 CB4HQ5 138539286 IC50 = 7.2 nM T32369 CIJQ46 140263405 IC50 = 77000 nM T32369 CGO4N2 155511166 IC50 = 16000 nM T32369 C8P0GC 155511168 IC50 = 12000 nM T32369 C7RU3H 155517494 IC50 = 27800 nM T32369 C9DJU6 155520844 IC50 = 1590 nM T32369 CQF48P 155525610 IC50 = 500 nM T32369 CNE5F2 155525938 IC50 = 103000 nM T32369 CT46MX 155533612 IC50 = 68000 nM T32369 CB8ZP7 155536386 IC50 = 298 nM T32369 C4DRB9 155536871 IC50 = 27400 nM T32369 CG0I1B 155537860 IC50 = 35000 nM T32369 COQ28E 155544636 IC50 > 809000 nM T32369 CV34YN 155551139 IC50 = 5000 nM T32369 CIA0T9 155554354 IC50 = 30000 nM T32369 C5OIB7 155555229 IC50 = 0.05012 nM T32369 CPES21 155564673 IC50 = 44000 nM T32369 CH68RB 155567110 IC50 = 9310 nM T32369 C4S6BL 155567739 IC50 = 65000 nM T32369 CK6PJ1 155567828 IC50 = 2990 nM T32369 C7YTS1 514095 EC50 > 250000 nM T32369 CW80LD 56659856 Ki = 2000 nM T32369 D05SSB 514100 Ki = 850 nM T32369 D0F3CO 3840 IC50 = 12300 nM T87554 D03ZBT 11626560 IC50 = 27 nM T87554 D04LKS 25126798 IC50 = 0.056 nM T87554 D04LVK 57379345 IC50 = 610 nM T87554 D07POC 176870 IC50 = 4000 nM T87554 D0E7PQ 5311 IC50 > 10000 nM T87554 D0EG1I 9926791 IC50 = 0.6 nM T87554 D0J9ZR 4477 IC50 = 10000 nM T87554 D0Y7IC 44205240 IC50 = 5.7 nM T87554 D00DRL 44137946 IC50 = 230 nM T87554 D00RYA 16750271 IC50 = 46 nM T87554 D02TUL 118115473 IC50 > 10000 nM T87554 D03LWG 53235510 IC50 = 2882 nM T87554 D04QWQ 59422203 Ki = 13 nM T87554 D05PCM 78323835 IC50 = 803 nM T87554 D05PZB 135398495 IC50 = 1 nM T87554 D06DMQ 59472121 Ki = 150 nM T87554 D06EIC 57928403 IC50 = 5 nM T87554 D07EHV 44814409 IC50 > 10000 nM T87554 D07HPJ 11476171 IC50 > 10000 nM T87554 D07JAG 58557659 IC50 = 120 nM T87554 D08DHN 67286591 Ki > 4000 nM T87554 D08HOM 46207586 IC50 > 10000 nM T87554 D0BI3N 44595079 IC50 = 6 nM T87554 D0D5ZJ 25062766 IC50 = 18 nM T87554 D0D8KQ 25127112 IC50 = 28 nM T87554 D0DK5X 135567296 IC50 = 23.1 nM T87554 D0DK8X 50922691 IC50 = 80 nM T87554 D0E3TC 44259 IC50 = 0.189 nM T87554 D0G8BM 16722836 IC50 = 3 nM T87554 D0G9AW 59473233 EC50 = 453 nM T87554 D0H2HZ 60194098 IC50 = 10000 nM T87554 D0MP0X 16659841 IC50 < 3 nM T87554 D0O0LS 25141092 IC50 = 40 nM T87554 D0O6WV 24794418 IC50 > 2000 nM T87554 D0P0KN 16739650 IC50 = 73 nM T87554 D0P1CV 46191454 IC50 > 10000 nM T87554 D0PN8H 46216796 IC50 = 1 nM T87554 D0R9IU 44462758 IC50 = 1750 nM T87554 D0S1XX 134821691 IC50 > 10000 nM T87554 D0S6TK 11213558 IC50 = 6 nM T87554 D0SG7B 49831257 IC50 = 2400 nM T87554 D03BNU 59604787 IC50 > 3500 nM T87554 D05PDI 46224913 Ki = 1 nM T87554 D0Y2PO 71770709 IC50 = 16600 nM T87554 D08DBE 10344820 Ki = 130 nM T87554 D0GZ7B 5328779 IC50 > 10000 nM T87554 D0T3ME 156422 IC50 > 30000 nM T87554 CBPM40 4878 IC50 > 50000000 nM T87554 CU68FI 78893 Ki = 3200 nM T87554 C6ZB4U 790291 Ki = 3000 nM T87554 CZJB27 817910 IC50 = 40900 nM T87554 CGQM48 869412 Ki = 1700 nM T87554 C0XL5P 951379 Ki > 3500 nM T87554 C7ZUW6 1246120 Ki = 2800 nM T87554 CI1B7L 1247281 Ki = 3200 nM T87554 CP6BI3 1481965 IC50 = 13000 nM T87554 C19-AUG 1927544 IC50 = 15000 nM T87554 CY35GB 2241431 IC50 = 6000 nM T87554 C4J8HV 2389948 IC50 = 13800 nM T87554 CWCH42 2786631 IC50 = 131000 nM T87554 C3F0GS 3120536 Ki = 1200 nM T87554 CD67OL 4250390 Ki > 3500 nM T87554 C6SNL5 4393251 Ki > 3500 nM T87554 CG9RD4 4448318 IC50 = 453 nM T87554 CK6L3O 5121684 Ki = 1700 nM T87554 CX01FS 5473838 IC50 = 60 nM T87554 CGYE97 6419765 IC50 = 61 nM T87554 C2OL7K 9796455 IC50 > 50000 nM T87554 CYA76E 9798589 IC50 > 100000 nM T87554 CQ89SE 9947841 IC50 = 600 nM T87554 CO70CQ 10107882 IC50 = 58 nM T87554 C7SFI1 10296883 IC50 > 10000 nM T87554 C7HBP6 10429593 IC50 > 10000 nM T87554 CBOP58 11293798 Ki > 10000 nM T87554 C26BZX 11362471 Ki > 10000 nM T87554 CWXB93 11397177 Ki > 10000 nM T87554 CT3VP7 11398307 IC50 = 25000000 nM T87554 CK83CN 11416425 IC50 = 40 nM T87554 CTG83F 11539329 Ki > 1500 nM T87554 CI0X1C 11567474 IC50 = 688 nM T87554 CMIL86 11590363 Ki > 1500 nM T87554 CDIW70 11597571 IC50 = 92 nM T87554 C0O3HT 11601868 IC50 = 790 nM T87554 CV8EU0 11612136 IC50 = 65 nM T87554 C9ZD2E 11626406 IC50 = 4891 nM T87554 CSM62L 11626920 IC50 = 29000 nM T87554 C9T6SC 11640926 Ki > 1500 nM T87554 CXG5W8 11646595 IC50 = 3 nM T87554 C5LHC6 11658542 IC50 = 145300 nM T87554 CP3U0W 11684933 IC50 > 8333 nM T87554 CU0E8O 11690457 Ki = 400 nM T87554 CB0AP2 11705863 Ki = 4400 nM T87554 CS36BH 11843159 IC50 = 240 nM T87554 C61TIL 11844913 IC50 = 333 nM T87554 C9JT4S 11847343 IC50 = 1721 nM T87554 CHR92S 11858109 IC50 = 3400 nM T87554 CNYB84 11951225 IC50 = 83 nM T87554 CASK85 11957393 IC50 = 5.9 nM T87554 C58YUH 11993785 IC50 = 30 nM T87554 CW53JC 11998038 Ki = 13 nM T87554 C0Y7MG 12083227 IC50 = 45000 nM T87554 C75SGK 12997800 IC50 = 3 nM T87554 CM9JA0 12997805 IC50 = 0.2 nM T87554 C0DUA7 15953425 IC50 = 4.4 nM T87554 C3JWA6 15953427 IC50 = 3.6 nM T87554 CWZM24 15953526 IC50 = 18 nM T87554 CFPW41 16007116 Ki > 1400 nM T87554 C12TIL 16058762 IC50 = 3 nM T87554 C1WJ2D 16070041 IC50 = 100 nM T87554 COIK65 16070059 IC50 = 150 nM T87554 C1U8XW 16109036 IC50 = 550 nM T87554 CGC34R 16118737 IC50 > 1030 nM T87554 CT8WS0 16126645 IC50 = 124 nM T87554 C5VPH9 16129448 IC50 = 57 nM T87554 CM32VW 16659676 IC50 = 4 nM T87554 CO3L1Q 16659677 IC50 = 10 nM T87554 CL38VY 16659680 IC50 < 3 nM T87554 C5LP4O 16659681 IC50 = 3 nM T87554 C0ECA7 16659682 IC50 = 4 nM T87554 CXYV28 16659836 IC50 < 3 nM T87554 CDTG08 16659837 IC50 < 3 nM T87554 C91SVD 16659838 IC50 < 3 nM T87554 CC10IO 16662069 IC50 = 4 nM T87554 CD1NT2 16662070 IC50 < 3 nM T87554 C19KHB 16664854 IC50 = 209 nM T87554 CO7E8C 16678106 IC50 = 104 nM T87554 C4TC3X 16722832 IC50 = 6 nM T87554 CY1E2N 16723801 IC50 = 133600 nM T87554 C4Q2TN 16739431 IC50 = 210 nM T87554 CWI96A 16739432 IC50 = 62 nM T87554 CSE35D 16739464 IC50 = 820 nM T87554 C20OFQ 16739508 IC50 = 330 nM T87554 CNFX02 16739511 IC50 = 82 nM T87554 C3AGL1 16739512 IC50 = 150 nM T87554 C0JTZ9 16739677 IC50 = 1700 nM T87554 C4IX1K 16739678 IC50 = 510 nM T87554 COZ7A1 16739706 IC50 = 1500 nM T87554 C0HB9T 16739709 IC50 = 1500 nM T87554 C0U8DY 16739710 IC50 = 120 nM T87554 COC6L0 16739741 IC50 > 10000 nM T87554 C1Z8WO 16739742 IC50 = 280 nM T87554 CPT2G0 16739743 IC50 > 10000 nM T87554 CPC5Q9 16739745 IC50 > 10000 nM T87554 CLY96T 16739777 IC50 = 90 nM T87554 C0TMW8 16739778 IC50 = 180 nM T87554 C1MAE7 16739807 IC50 > 10000 nM T87554 C9H8XT 16739808 IC50 > 10000 nM T87554 CC5UB1 16739809 IC50 = 3300 nM T87554 CQ43TS 16739810 IC50 = 48 nM T87554 CJCN32 16739811 IC50 > 10000 nM T87554 CDK6A4 16739812 IC50 = 120 nM T87554 CE0I5O 16739835 IC50 = 160 nM T87554 C4C7DF 16739839 IC50 = 49 nM T87554 C20BPQ 16739840 IC50 = 56 nM T87554 CE1XT6 16739866 IC50 = 1350 nM T87554 C8JBR9 16739867 IC50 = 220 nM T87554 C1VG0U 16739870 IC50 = 62 nM T87554 C2Z4DB 16739901 IC50 = 110 nM T87554 C1UFH7 16739902 IC50 = 220 nM T87554 C7DFM1 16739903 IC50 = 1600 nM T87554 CHX86I 16739904 IC50 = 720 nM T87554 CCP56J 16739905 IC50 = 90 nM T87554 CP9C6B 16739918 IC50 = 100 nM T87554 CJB7M2 16739919 IC50 = 50 nM T87554 C2WNB4 16739920 IC50 = 50 nM T87554 CQ64XI 16739921 IC50 = 170 nM T87554 C9MT8U 16739933 IC50 = 140 nM T87554 CM3UF8 16739935 IC50 = 1100 nM T87554 CFEP56 16739948 IC50 = 260 nM T87554 CKE6V9 16739949 IC50 = 230 nM T87554 C23KZR 16739951 IC50 > 10000 nM T87554 C6GJ5Q 16739952 IC50 = 44 nM T87554 CFRU87 16739965 IC50 = 150 nM T87554 C9OQ1G 16750272 IC50 = 220 nM T87554 CW2SY5 16750291 IC50 = 7.3 nM T87554 CIX7U2 16750304 IC50 = 67 nM T87554 C6A3XS 16750306 IC50 = 17 nM T87554 CB2TK1 16750327 IC50 = 110 nM T87554 CH4O1C 16750328 IC50 = 290 nM T87554 C90MJD 16750331 IC50 = 930 nM T87554 C9MNP2 17549086 IC50 = 8900 nM T87554 CL9BQ6 17748275 IC50 = 1746 nM T87554 C6UAZ0 20820292 IC50 >= 10000 nM T87554 CE7K3W 23532567 IC50 > 10000 nM T87554 C1O6ME 23581858 IC50 = 210 nM T87554 C9WRS3 23581859 IC50 = 52 nM T87554 CYH2Z8 23582563 IC50 = 210 nM T87554 CWEC02 23582564 IC50 = 49 nM T87554 CRO1A2 23582565 IC50 = 230 nM T87554 CD7M2U 23582566 IC50 = 230 nM T87554 CZF6W3 23582567 IC50 = 68 nM T87554 CXZ87O 23582568 IC50 = 190 nM T87554 C6O5JX 23582570 IC50 = 17 nM T87554 CHS9L8 23582639 IC50 = 74 nM T87554 C53OJF 23582642 IC50 = 83 nM T87554 CM9A4G 23582643 IC50 = 51 nM T87554 CBC4Y7 23582701 IC50 = 18 nM T87554 CUY98W 23585560 IC50 = 19 nM T87554 CD0R9O 24699546 Ki = 3200 nM T87554 C7YG1N 24759534 IC50 = 2400 nM T87554 CAJ4T2 24762205 IC50 > 10000 nM T87554 CQNP54 24764449 IC50 = 25000 nM T87554 CFS2M7 24798487 Ki = 59.7 nM T87554 CLBP72 24798571 IC50 = 138 nM T87554 CX1U4S 24800423 IC50 = 15 nM T87554 C4T0DG 24800602 IC50 = 840 nM T87554 CH3ZG7 24800604 IC50 = 440 nM T87554 CBA02Y 24800776 IC50 = 8 nM T87554 C3UFG1 24801129 IC50 = 5 nM T87554 CVR8S1 24801650 IC50 = 110 nM T87554 CV5RP8 24809765 IC50 = 695 nM T87554 C29ANE 24809801 IC50 = 615 nM T87554 C59FKG 24860777 IC50 = 900 nM T87554 CL0O9E 24877325 IC50 = 12.6 nM T87554 CY0P4X 24877326 IC50 = 3.6 nM T87554 C7R4YV 24877438 IC50 = 6.9 nM T87554 C5G4BY 24877439 IC50 = 4.2 nM T87554 C5NXH3 24877440 IC50 = 6.5 nM T87554 CJ4Z0K 24877791 IC50 = 5.1 nM T87554 CQUH61 24877795 IC50 = 11.1 nM T87554 CO5RV2 24878018 IC50 = 4.4 nM T87554 CH3Q1D 24878130 IC50 = 39.6 nM T87554 CFK2B9 24882503 IC50 > 10000 nM T87554 CWV98O 24899557 IC50 = 1600 nM T87554 CLZ23U 24951610 IC50 = 21000 nM T87554 C5S7XA 24958852 IC50 = 41 nM T87554 CJ68PR 24958855 IC50 = 100 nM T87554 CZ18IU 24963047 IC50 = 78 nM T87554 CS3Q8B 24995659 Ki > 4000 nM T87554 CT07ZW 25030805 IC50 = 3 nM T87554 CHLC27 25052652 IC50 = 25 nM T87554 C7W6FX 25059112 IC50 = 8 nM T87554 CD0T4Z 25059626 IC50 = 116 nM T87554 CD4TJ7 25059891 IC50 = 374 nM T87554 CE9N8F 25060146 IC50 = 10 nM T87554 C3Y7SB 25060677 IC50 = 186 nM T87554 CWZH04 25060922 IC50 = 41 nM T87554 C7VPB2 25060927 IC50 = 30 nM T87554 C25NMK 25061435 IC50 = 163 nM T87554 CLH91O 25061438 IC50 = 326 nM T87554 CF3Z0Q 25061949 IC50 = 113 nM T87554 CF3QE4 25061950 IC50 = 549 nM T87554 C2BEQ3 25062226 IC50 = 132 nM T87554 CSVH95 25062228 IC50 = 303 nM T87554 C9KY0J 25062498 IC50 = 65 nM T87554 CG4U2Y 25062765 IC50 = 545 nM T87554 C2FI3E 25062767 IC50 = 533 nM T87554 CVI87D 25063021 IC50 = 52 nM T87554 C4JO2C 25063023 IC50 = 298 nM T87554 C3VIR1 25063025 IC50 = 166 nM T87554 C2KY1G 25094210 IC50 > 10000 nM T87554 C2H4VG 25096016 IC50 = 1 nM T87554 C9YVJ0 25096019 IC50 = 75 nM T87554 C8DTP7 25096020 IC50 = 27 nM T87554 CQA4V6 25096276 IC50 = 53 nM T87554 C40GWA 25096277 IC50 = 1115 nM T87554 CF7TP1 25096279 IC50 = 750 nM T87554 C2V4IM 25096280 IC50 = 100 nM T87554 C05XPV 25096532 IC50 = 4100 nM T87554 CV8PC6 25097027 IC50 = 540 nM T87554 CUB4W5 25102935 IC50 = 5 nM T87554 CM0O7N 25102936 IC50 < 3 nM T87554 C3PKV4 25102938 IC50 < 3 nM T87554 CNQ07G 25103042 IC50 = 6 nM T87554 C09PMH 25103279 IC50 = 3 nM T87554 C1V7QM 25103281 IC50 = 4 nM T87554 COP15B 25103284 IC50 = 17 nM T87554 CP8GU7 25104502 IC50 = 5 nM T87554 C7EK6V 25104503 IC50 = 6 nM T87554 C63ADF 25104611 IC50 = 37 nM T87554 CPM6S0 25104740 IC50 < 3 nM T87554 CJW1T2 25104741 IC50 = 3 nM T87554 CON1U6 25110598 IC50 = 7.5 nM T87554 C0JYA9 25123154 IC50 = 72 nM T87554 C56JVD 25123155 IC50 = 13 nM T87554 CZM6Q2 25123472 IC50 = 5.1 nM T87554 C3IA7V 25123474 IC50 = 120 nM T87554 C6V4NB 25123475 IC50 = 20 nM T87554 C0KOU6 25123487 IC50 = 34 nM T87554 CFK89A 25123806 IC50 = 14 nM T87554 C3RMN9 25123807 IC50 = 20 nM T87554 C5GO3T 25123808 IC50 = 195 nM T87554 C0W8IC 25124143 IC50 = 20 nM T87554 C61WOA 25127137 IC50 = 65 nM T87554 CTPV83 25127138 IC50 = 270 nM T87554 C8ASE3 25127139 IC50 = 398 nM T87554 CY32NR 25127140 IC50 = 178 nM T87554 C2K6UF 25127142 IC50 = 161 nM T87554 C6O4ES 25127144 IC50 = 227 nM T87554 CVQT51 25127461 IC50 = 146 nM T87554 C3UM5H 25127784 IC50 = 891 nM T87554 CF2W8C 25127785 IC50 = 16 nM T87554 C4WFL0 25128110 IC50 = 42 nM T87554 CWD72X 25128951 Ki = 1.6 nM T87554 CM86LX 25128955 Ki = 4200 nM T87554 C56TUK 25128956 Ki = 71 nM T87554 CXJ02U 25129311 Ki = 3100 nM T87554 CHD16N 25129655 Ki = 2 nM T87554 CS1FT7 25130358 Ki = 2400 nM T87554 C6G4DB 25130691 Ki = 2400 nM T87554 C6PAD3 25130693 Ki = 4 nM T87554 C6PXJ0 25130695 Ki = 1500 nM T87554 C9N6KS 25131017 Ki = 200 nM T87554 CND06Y 25131018 Ki = 130 nM T87554 C7GR4S 25131021 Ki = 1300 nM T87554 CF7PV8 25131681 Ki = 56 nM T87554 CFZ23Q 25132021 Ki = 280 nM T87554 CM9O4G 25132023 Ki = 210 nM T87554 C7AY6L 25132025 Ki = 1000 nM T87554 CE20BM 25132384 Ki = 1100 nM T87554 CZO81Q 25132387 Ki = 2000 nM T87554 CXI03Y 25132388 Ki = 3400 nM T87554 C9OCM7 25132389 Ki = 1700 nM T87554 C2NXD1 25132390 Ki = 750 nM T87554 CAL6Y5 25132729 Ki = 490 nM T87554 CE52HX 25132730 Ki = 2900 nM T87554 CS7TM1 25132733 Ki = 210 nM T87554 C9DYQ1 25133399 Ki = 220 nM T87554 COV8Z0 25143021 IC50 > 10000 nM T87554 C6BWZ8 25145145 IC50 > 100 nM T87554 C78YWA 25145716 IC50 > 500 nM T87554 CI0E2L 25154395 IC50 = 18 nM T87554 CL1W5D 25154436 IC50 = 14 nM T87554 CB21XV 25164469 Ki = 91 nM T87554 CUX83H 25164675 Ki = 351 nM T87554 C1H7BF 25164677 Ki = 482 nM T87554 C6SD2A 25165081 Ki > 1453 nM T87554 C67TVH 25165085 Ki = 1282 nM T87554 C8J4KL 25165278 Ki = 16 nM T87554 CRJ6M7 25165279 Ki > 1450 nM T87554 C7RBX0 25165280 Ki > 1450 nM T87554 CPEY29 25165481 Ki > 1450 nM T87554 C70DRX 25165482 Ki > 1450 nM T87554 CE8D1W 25165860 Ki = 1453 nM T87554 C6VZU2 25165861 Ki = 284 nM T87554 CT94MS 25166059 Ki > 1453 nM T87554 C5BM7F 25166250 Ki = 1450 nM T87554 C2D3FP 25167078 Ki > 1450 nM T87554 C8GL6I 25169133 IC50 < 3 nM T87554 C1G5JU 25169403 IC50 = 346 nM T87554 CZ28ES 25171661 IC50 < 3 nM T87554 CBIA60 25171662 IC50 = 4 nM T87554 C6ZTG4 25171663 IC50 < 3 nM T87554 CQH5N9 25171664 IC50 = 3 nM T87554 CQ04LW 25171665 IC50 < 3 nM T87554 CU9KV5 25171666 IC50 = 3 nM T87554 C0SE7H 25171874 IC50 < 3 nM T87554 C1YH8L 25171876 IC50 < 3 nM T87554 CC60NT 25171877 IC50 = 10 nM T87554 C8O1ZJ 25172085 IC50 < 3 nM T87554 CG6J5X 25172086 IC50 < 3 nM T87554 C0PX8V 25172087 IC50 = 33 nM T87554 C6UQG4 25181422 IC50 = 39 nM T87554 CX7CP9 25195487 IC50 = 200 nM T87554 CNG96H 25210579 IC50 > 10000 nM T87554 C0ZXH7 25236808 Ki = 2000 nM T87554 CC71QJ 27666048 IC50 > 100000 nM T87554 CT7X8Y 27700054 Ki > 3500 nM T87554 CW3QI4 42600633 Ki = 82.6 nM T87554 C92QDU 42611189 Ki = 86 nM T87554 CY4LG8 42622934 IC50 = 0.8 nM T87554 CAO2T4 42634832 Ki = 270 nM T87554 C57VJY 42635854 IC50 = 0.4 nM T87554 CP8RA7 42635855 IC50 = 1 nM T87554 C05BWT 42635901 IC50 = 1 nM T87554 CO9Y8F 42635906 IC50 = 11 nM T87554 CN1TI5 42635944 IC50 = 1 nM T87554 C5I9XW 42635949 IC50 = 2 nM T87554 CT63QC 42635982 IC50 = 95 nM T87554 CY5E4B 42635983 IC50 = 2 nM T87554 C8V6IK 42635984 IC50 = 3 nM T87554 C63HQD 42636016 IC50 = 2 nM T87554 C34DCR 42636018 IC50 = 2 nM T87554 CTOQ08 42636019 IC50 = 2 nM T87554 CU8MO6 42641406 IC50 = 6 nM T87554 CCB1E9 44124695 IC50 > 100000 nM T87554 CQI60M 44158549 IC50 = 6900 nM T87554 CBAN65 44158553 IC50 = 52 nM T87554 CH6OL2 44158658 IC50 = 3.4 nM T87554 CHD5N8 44158660 IC50 = 7.8 nM T87554 CU07NR 44158886 IC50 = 11 nM T87554 CLK7R8 44159000 IC50 = 0.5 nM T87554 CD0YP3 44159001 IC50 = 0.6 nM T87554 CQ8FJ4 44159590 IC50 = 3000 nM T87554 CY67LR 44159594 IC50 = 1.4 nM T87554 CZF1B5 44159711 IC50 = 1500 nM T87554 CQW4F1 44159839 IC50 = 34 nM T87554 CBK83A 44159959 IC50 = 22 nM T87554 CEF0X4 44159962 IC50 = 36 nM T87554 CBZ09W 44160079 IC50 = 560 nM T87554 C1ZY4N 44160207 IC50 = 0.2 nM T87554 CB0O2A 44186880 Ki = 1453 nM T87554 C9K7OP 44186882 Ki = 756 nM T87554 CX0ZU8 44186885 Ki = 1453 nM T87554 CNGV37 44189584 Ki > 1450 nM T87554 CIT2A7 44192904 IC50 = 76.7 nM T87554 C8KNA3 44219632 Ki > 4000 nM T87554 C0VIX4 44219633 Ki = 2400 nM T87554 CZB49P 44419474 IC50 = 19 nM T87554 CI9GX4 44419475 IC50 = 17 nM T87554 CAT2U0 44419478 IC50 = 68 nM T87554 CC36WM 44419481 IC50 = 113 nM T87554 C6BWA2 44419485 IC50 = 59 nM T87554 CXW0D5 44419491 IC50 = 4 nM T87554 CZY28V 44419492 IC50 = 8 nM T87554 CCM3W5 44419493 IC50 = 16 nM T87554 CG2R1T 44419498 IC50 = 51 nM T87554 C40WFE 44419499 IC50 = 153 nM T87554 CNZJ15 44419502 IC50 = 20 nM T87554 C5DL8E 44419515 IC50 > 10000 nM T87554 CMVY72 44419516 IC50 = 167 nM T87554 CNT03L 44419522 IC50 = 7218 nM T87554 CH46CM 44419523 IC50 = 51 nM T87554 CO20LA 44419524 IC50 = 12 nM T87554 C3CBQ4 44419526 IC50 = 49 nM T87554 C4XIY6 44419527 IC50 > 10000 nM T87554 CGH30Q 44419528 IC50 = 77 nM T87554 C42FJP 44419532 IC50 > 10000 nM T87554 C0FKV6 44419533 IC50 = 18 nM T87554 CXG7H4 44419544 IC50 = 56 nM T87554 CI2BL7 44419547 IC50 = 141 nM T87554 C2T5AQ 44419548 IC50 = 29 nM T87554 CT19AN 44419556 IC50 = 28 nM T87554 CE6T5F 44419559 IC50 = 7 nM T87554 CQ0Y6P 44432177 IC50 = 11 nM T87554 CSRD60 44432179 IC50 = 6 nM T87554 C1DZ5C 44432180 IC50 = 19 nM T87554 CWBI39 44432182 IC50 = 55 nM T87554 C73SGA 44432183 IC50 = 42 nM T87554 CA92GM 44432184 IC50 = 21 nM T87554 CTDI23 44432185 IC50 = 53 nM T87554 CI9NY3 44432187 IC50 = 25 nM T87554 CGFT15 44432188 IC50 = 222 nM T87554 CT0D6O 44432189 IC50 = 132 nM T87554 CFK94T 44432190 IC50 = 359 nM T87554 C3TG1J 44432191 IC50 = 323 nM T87554 CBO5P0 44432192 IC50 = 298 nM T87554 C2S8ZC 44432193 IC50 = 1860 nM T87554 CYH6P3 44520205 IC50 > 10000 nM T87554 CW2P1N 44555004 Ki = 1.7 nM T87554 C96QIW 44555963 Ki = 2 nM T87554 CP5M6H 44556110 Ki = 1.1 nM T87554 CQ18YJ 44556112 Ki = 0.6 nM T87554 C3VRO9 44557921 IC50 > 10000 nM T87554 COR3N9 44560358 IC50 = 572 nM T87554 CA69DI 44570386 IC50 = 9300 nM T87554 C8A2ZJ 44570387 IC50 = 1950 nM T87554 C0S8WJ 44570388 IC50 = 28600 nM T87554 CR7T0U 44570389 IC50 = 320 nM T87554 C5YL2S 44570390 IC50 = 370 nM T87554 CVC6A3 44570391 IC50 = 740 nM T87554 C5A8CV 44570392 IC50 = 5800 nM T87554 C6B3XH 44570434 IC50 = 8580 nM T87554 CS6MF4 44570435 IC50 = 3550 nM T87554 C45TSL 44570436 IC50 = 1950 nM T87554 CCRL12 44570437 IC50 = 3900 nM T87554 C0EC7O 44570438 IC50 = 1570 nM T87554 CF1Y6E 44570474 IC50 = 1110 nM T87554 C1JSB3 44570475 IC50 = 330 nM T87554 CRGC97 44570476 IC50 = 1220 nM T87554 C9B8UC 44570477 IC50 = 770 nM T87554 C8KQ9B 44605608 Ki = 210 nM T87554 C63WNF 44610370 IC50 = 1010 nM T87554 CT7V9E 44610371 IC50 = 319 nM T87554 CL40ZN 44610523 IC50 = 175 nM T87554 C6QT0J 44622837 IC50 > 1000 nM T87554 C9AVD2 44624425 Ki = 1.6 nM T87554 CKUA84 44626045 IC50 > 30000 nM T87554 C2SLI6 44631938 IC50 = 18 nM T87554 C4K8BX 45267171 IC50 = 33500 nM T87554 C25VIM 45267176 IC50 = 16900 nM T87554 C36DGY 45272290 IC50 > 40000 nM T87554 COT0W8 45272300 IC50 = 5100 nM T87554 CC79UA 45273165 IC50 > 40000 nM T87554 CNR8G6 45273175 IC50 > 40000 nM T87554 C4J5XF 45275254 IC50 = 4 nM T87554 CZ7T8F 45275363 IC50 = 15 nM T87554 CB58EO 45275368 IC50 = 27 nM T87554 CU3AD0 45275473 IC50 = 12 nM T87554 C7KMO9 45275580 IC50 = 3 nM T87554 CFN17Z 45280146 IC50 = 1.1 nM T87554 CA23WL 45280210 IC50 = 6 nM T87554 C96HCQ 45375954 IC50 = 56 nM T87554 CQ3KO2 45375955 IC50 = 1.2 nM T87554 C5G2MN 45375956 IC50 = 5 nM T87554 C6OX0V 45375974 IC50 < 3 nM T87554 C0QP2U 45483928 Ki = 260 nM T87554 CS7RO0 45483929 Ki = 480 nM T87554 CXF92W 45486106 IC50 = 200 nM T87554 CZXL23 45486109 IC50 = 44 nM T87554 CF8JM7 45486113 IC50 = 6500 nM T87554 CIE6V0 45486118 IC50 = 84 nM T87554 CV59GT 45486119 IC50 = 260 nM T87554 C9E0MS 45486120 IC50 = 4.7 nM T87554 C07DPA 45486121 IC50 = 4 nM T87554 CR7T9D 45486124 IC50 = 210 nM T87554 C7QK0X 45486129 IC50 = 880 nM T87554 CY36ZX 45486130 IC50 = 70 nM T87554 C04ZHY 45486136 IC50 = 50 nM T87554 C5SA2N 45486137 IC50 = 190 nM T87554 C91VMT 45486138 IC50 = 25 nM T87554 CLN7F0 45486139 IC50 = 3.1 nM T87554 C8RNJ5 45486142 IC50 = 270 nM T87554 C9FQJ4 45486147 IC50 = 87 nM T87554 CPM6O9 45486148 IC50 = 130 nM T87554 CX0HO6 45486156 IC50 < 3 nM T87554 CYZ13M 45486157 IC50 = 907 nM T87554 CZMD28 45486158 IC50 = 160 nM T87554 CMXY69 45486159 IC50 = 4.6 nM T87554 CA0O3Q 45486163 IC50 = 20 nM T87554 C5U1LS 45486164 Ki = 7 nM T87554 CN6G7A 45486168 IC50 = 4 nM T87554 CT9OP5 45486169 IC50 = 4666 nM T87554 C7D4GB 45486170 IC50 = 21 nM T87554 CET79H 45493316 IC50 = 110 nM T87554 CND6H4 46176417 IC50 = 120 nM T87554 CE45XW 46208354 IC50 = 4.9 nM T87554 CUHB49 46208355 IC50 = 4.1 nM T87554 CW38GO 46208357 IC50 = 5.5 nM T87554 C43COY 46208358 IC50 = 3.2 nM T87554 CE4Q7D 46208596 IC50 = 5.3 nM T87554 CM9UN7 46208601 IC50 = 1.1 nM T87554 CH7JB4 46209051 IC50 = 3.5 nM T87554 CY3HW5 46224684 IC50 > 10000 nM T87554 CLOZ21 46224796 Ki = 0.5 nM T87554 C9O2RG 46224797 Ki = 0.6 nM T87554 C9BET8 46224835 Ki = 13 nM T87554 C6TU1W 46224836 Ki = 42 nM T87554 C03MZI 46224837 Ki = 3 nM T87554 C9RGH2 46224876 Ki = 2100 nM T87554 C0C9IJ 46224910 Ki > 5000 nM T87554 CLPV83 46224911 Ki > 5000 nM T87554 CM8Z4P 46224912 Ki = 3800 nM T87554 CA4V3E 46224936 Ki = 1 nM T87554 CJ0P5D 46224938 Ki = 400 nM T87554 CVZ80Y 46224939 Ki = 4500 nM T87554 CG3SZ2 46224940 Ki > 5000 nM T87554 C3DJ5Q 46224970 Ki > 5000 nM T87554 C0NFE6 46224971 Ki = 29 nM T87554 C3R0EQ 46224972 Ki = 630 nM T87554 CI83TA 46224997 Ki = 34 nM T87554 C4VU8O 46224998 Ki = 3800 nM T87554 C86GDI 46225269 Ki = 2100 nM T87554 C9AJP4 46225270 Ki = 460 nM T87554 CV37ID 46225315 Ki = 1800 nM T87554 C1Z0JB 46225316 Ki = 370 nM T87554 CG6Y3N 46234403 IC50 = 234 nM T87554 C3JW8A 46234405 IC50 = 226 nM T87554 CWN3M0 46234565 EC50 = 2045 nM T87554 CLTU68 46234566 IC50 = 78 nM T87554 C5YH1F 46235625 IC50 = 47 nM T87554 CWLU63 46235938 IC50 = 181 nM T87554 CC25DT 46235942 IC50 = 7 nM T87554 CZ7J6K 46236109 IC50 = 48 nM T87554 C26NQY 46236112 IC50 = 92 nM T87554 C1S4LH 46398810 IC50 = 7.3 nM T87554 CG71EF 46832441 IC50 = 2 nM T87554 C1LNX9 46832443 IC50 = 5.5 nM T87554 CCK54P 46852509 IC50 = 85 nM T87554 CC57FP 46852510 IC50 = 8.9 nM T87554 C31UXV 46852812 IC50 = 13 nM T87554 COTJ39 46863083 IC50 = 13000 nM T87554 C35AIH 46865430 IC50 = 5 nM T87554 C2EK4B 46865431 IC50 = 5 nM T87554 CMZ0R3 46865529 IC50 = 4.3 nM T87554 C3B2NL 46865530 IC50 = 6.8 nM T87554 CC2O9R 46865656 IC50 = 1584.89 nM T87554 CJ3NV8 46865657 IC50 = 8 nM T87554 CQB16A 46872415 Ki = 3200 nM T87554 CLS29B 46872626 IC50 > 10000 nM T87554 C0AU7R 46879420 IC50 = 28 nM T87554 CUVG95 46879421 IC50 = 1550 nM T87554 CRZM17 46879422 IC50 = 170 nM T87554 CER6X5 46879423 IC50 = 97 nM T87554 C7O1AZ 46879483 IC50 = 500 nM T87554 C2DU1O 46879484 IC50 = 95 nM T87554 CB31AL 46879485 IC50 = 285 nM T87554 C5URZ1 46879545 IC50 = 840 nM T87554 C3LEW4 46879546 IC50 = 7000 nM T87554 CKI4M6 46880119 IC50 = 3250 nM T87554 CU8KB7 46880120 IC50 = 1800 nM T87554 C47OXF 46880121 IC50 = 560 nM T87554 CK87XC 46880122 IC50 = 3400 nM T87554 CC3Y7B 46880193 IC50 = 393 nM T87554 C0GS1C 46880194 IC50 = 470 nM T87554 CV9IL3 46880195 IC50 = 1000 nM T87554 C0M5ND 46880196 IC50 = 270 nM T87554 C60UAN 46880197 IC50 = 320 nM T87554 C5NZ8R 46880686 IC50 = 150 nM T87554 CZ79VE 46880687 IC50 = 8 nM T87554 C0YNH6 46880737 IC50 < 3 nM T87554 CGO7C5 46880738 IC50 = 14 nM T87554 C75ZTG 46880739 IC50 = 39 nM T87554 C9T7WL 46880784 IC50 = 8 nM T87554 CSV4G2 46880785 IC50 = 5 nM T87554 CS6W4P 46882359 IC50 = 467 nM T87554 CF5B9A 46882360 IC50 = 322 nM T87554 CX4UK2 46882361 IC50 = 202 nM T87554 C5FNK6 46882409 IC50 = 83 nM T87554 CN8OR4 46882410 IC50 = 81 nM T87554 CEI25D 46882411 IC50 = 33 nM T87554 CJZ8H9 46882412 IC50 = 16 nM T87554 C6Z4KW 46882470 IC50 = 6 nM T87554 CH0Y5K 46882471 IC50 = 11 nM T87554 C70LVA 46882472 IC50 = 8 nM T87554 CP1BH3 46882539 IC50 = 12 nM T87554 CQR25C 46882540 IC50 = 9 nM T87554 CVTO81 46882541 IC50 = 16 nM T87554 CQ6T0Y 46882542 IC50 = 14 nM T87554 COV4E6 46882589 IC50 = 18 nM T87554 CDG2N8 46882590 IC50 = 2 nM T87554 C0UX2M 46882591 IC50 = 4 nM T87554 CN0I6Z 46882592 IC50 = 6 nM T87554 CZ7A9N 46882802 IC50 = 69 nM T87554 CCK7H2 46882803 IC50 = 47 nM T87554 C9MW2L 46885052 IC50 = 4200 nM T87554 C69HUW 46885053 IC50 = 101 nM T87554 CASL67 46885231 IC50 = 685 nM T87554 CEU6O4 46885232 IC50 = 501 nM T87554 CE27LI 46885233 IC50 = 7.1 nM T87554 CB8LN4 46885234 IC50 = 13 nM T87554 CMX7U6 46885289 IC50 = 12.5 nM T87554 CB1ZN5 46885290 IC50 = 3.1 nM T87554 C2O8RZ 46886323 IC50 > 1000 nM T87554 C60GAV 46929544 IC50 > 8000 nM T87554 CP34VL 46929748 IC50 > 1000 nM T87554 CJ2E9Q 46929857 IC50 > 25000 nM T87554 CCN08S 46934144 IC50 = 106700 nM T87554 CT7EY8 49817363 IC50 = 330 nM T87554 CBP75U 49838138 IC50 = 0.9 nM T87554 CMKB24 49838268 IC50 = 3 nM T87554 CF0UM2 49838516 IC50 = 0.64 nM T87554 CTJX98 49838518 IC50 = 1.4 nM T87554 CSE4K3 49838775 IC50 = 1.27 nM T87554 CB34CO 49839441 Ki = 35 nM T87554 C2DGY0 49839445 Ki > 3500 nM T87554 C06MKW 49839561 Ki = 27.6 nM T87554 CT3SH4 49839838 IC50 = 3 nM T87554 CF91RS 49843531 IC50 > 10000 nM T87554 C7A6IZ 49850211 EC50 > 20000 nM T87554 C57FQH 49856318 IC50 = 790 nM T87554 C70QSD 49856319 IC50 = 510 nM T87554 C24SMN 49856320 IC50 = 1440 nM T87554 CHK7D3 49856321 IC50 = 480 nM T87554 CK4LJ5 49856703 Ki = 770 nM T87554 CZVU24 49856845 Ki = 0.3 nM T87554 C9J7LZ 49857227 Ki = 7.1 nM T87554 CS72TM 49859752 IC50 = 1.8 nM T87554 CK5TH3 50906783 EC50 = 2800 nM T87554 CA0WR3 50914031 IC50 = 250 nM T87554 CQE9D1 50925411 IC50 = 578 nM T87554 C64HTN 50925513 IC50 = 1 nM T87554 C2Y6QS 50938552 IC50 > 10000 nM T87554 CF26MU 50991562 IC50 = 33 nM T87554 CHS63D 50993724 IC50 < 3 nM T87554 C2SKV4 50993725 IC50 = 9 nM T87554 CKN2H7 50993726 IC50 = 16 nM T87554 CMH3A2 50993881 IC50 < 3 nM T87554 C20VEP 50994284 IC50 > 10000 nM T87554 CI1L0M 50994285 IC50 = 4700 nM T87554 C7ZWT8 50994286 IC50 = 9150 nM T87554 C6VNE1 50994366 IC50 = 1444 nM T87554 CSEZ73 50994367 IC50 > 10000 nM T87554 C1R8ZI 50995341 IC50 = 129 nM T87554 C53NRD 50995522 IC50 = 180 nM T87554 CAZQ43 51003133 IC50 > 1000 nM T87554 CWKS75 51003514 IC50 = 1 nM T87554 C9NYP4 51036677 IC50 > 10000 nM T87554 C4WRY3 51037112 IC50 > 10000 nM T87554 CRI28Z 51037948 IC50 > 10000 nM T87554 CDU4Q5 51346827 Ki = 898 nM T87554 CXA03W 52920796 IC50 > 100 nM T87554 CEQN27 52936621 Ki = 370 nM T87554 C1PLW9 52941200 IC50 = 1400 nM T87554 CA9DE6 52941228 IC50 > 10000 nM T87554 CR2QD0 52941284 IC50 = 8350 nM T87554 C1T5EH 52942437 IC50 > 10000 nM T87554 C54UKL 52942449 IC50 = 3940 nM T87554 CO8W1R 52942701 IC50 = 55 nM T87554 CY20GZ 52942702 IC50 = 274 nM T87554 CEPS91 52943663 IC50 = 5000 nM T87554 C2IQ5B 52943672 IC50 > 10000 nM T87554 CMP9W8 52944434 IC50 = 139 nM T87554 CTN0C3 52944839 IC50 > 10000 nM T87554 CXG0B3 52946111 IC50 = 3157 nM T87554 CN2Q0G 52946313 IC50 = 14 nM T87554 CT2U3E 52947304 IC50 = 2500 nM T87554 CU49PE 52947324 IC50 = 11500 nM T87554 C1QWK5 52947390 IC50 = 512 nM T87554 CY42JP 52947547 IC50 = 200 nM T87554 C7S8TB 52948490 IC50 = 29000 nM T87554 CQY9D0 52948526 IC50 = 2110 nM T87554 C8TC3P 52948550 IC50 = 2500 nM T87554 CIM43G 52948562 IC50 > 10000 nM T87554 CWG31A 52948678 IC50 = 4 nM T87554 CQ87RP 52949754 IC50 = 11800 nM T87554 CNW53F 52949761 IC50 = 630 nM T87554 C6VHI5 52949798 IC50 = 26 nM T87554 C2XNP3 53024548 IC50 = 12200 nM T87554 CR36JQ 53232414 IC50 = 115300 nM T87554 C93WOC 53232452 IC50 < 3 nM T87554 C6OTY5 53251320 IC50 = 11000 nM T87554 CZ71UE 53316996 IC50 = 190 nM T87554 CE5Y7P 53316997 IC50 = 110 nM T87554 CH13DY 53316998 IC50 = 22 nM T87554 CXO42U 53317010 IC50 = 5.3 nM T87554 C3HT4Y 53317607 IC50 = 2 nM T87554 CH3Y2L 53317729 IC50 = 14000 nM T87554 C8KXF6 53317730 IC50 = 22 nM T87554 CE8OY2 53317913 IC50 > 100 nM T87554 CI8PJ6 53318277 IC50 = 2700 nM T87554 C7T2RG 53318278 IC50 = 2.2 nM T87554 C4RBZ8 53318283 IC50 = 3.5 nM T87554 C7D4IR 53318284 IC50 = 4.6 nM T87554 CZS8K4 53319042 Ki = 791 nM T87554 CGRX02 53319638 IC50 = 31 nM T87554 C6QP8W 53319646 IC50 = 7.3 nM T87554 C8OAH1 53319647 IC50 = 0.6 nM T87554 C5ZT4W 53319648 IC50 = 2.4 nM T87554 CUD21V 53320263 Ki = 644 nM T87554 C76DUB 53320946 IC50 = 4.8 nM T87554 C0XZA6 53320947 IC50 = 1.2 nM T87554 CF4LM9 53321614 IC50 = 2.8 nM T87554 CFHD02 53322268 IC50 = 59 nM T87554 CESA85 53323614 Ki = 281 nM T87554 C39GZV 53323629 IC50 = 1.1 nM T87554 C2W9OA 53324451 IC50 > 10000 nM T87554 C8M9WN 53324904 IC50 = 4.5 nM T87554 CU6W1L 53324912 IC50 = 2.1 nM T87554 CB94UN 53326192 IC50 = 9.3 nM T87554 CVY30S 53326193 IC50 = 3 nM T87554 CEF6L2 53326206 IC50 = 0.9 nM T87554 CQS1R8 53341008 Ki = 28 nM T87554 CNPM14 53341082 IC50 > 3000 nM T87554 C4BM5W 53341107 Ki = 12 nM T87554 CZKQ72 53341161 Ki = 53 nM T87554 CN59SH 53341248 Ki = 10 nM T87554 CB83XH 53341368 Ki = 56 nM T87554 CD2CH6 53341413 Ki = 40 nM T87554 CGP23R 53341457 Ki = 1.2 nM T87554 C0SWH5 53348216 IC50 > 40000 nM T87554 C8ZRE3 53356518 IC50 = 3068 nM T87554 C95JTI 53373594 Ki = 6.5 nM T87554 C8NA4L 53384644 IC50 > 30000 nM T87554 C56TYK 53385837 IC50 = 121.6 nM T87554 CNLM53 53385838 IC50 = 123.1 nM T87554 C1XE2K 53385938 IC50 = 345.4 nM T87554 C37JTE 53385939 IC50 = 37 nM T87554 CV92IB 53386254 IC50 = 18 nM T87554 CU6QF7 53386309 IC50 < 0.6 nM T87554 CYU0R4 53386418 IC50 = 0.5 nM T87554 C7RM6Q 53386421 IC50 < 0.3 nM T87554 CEN91X 53389820 IC50 = 231.2 nM T87554 C24FQU 53465297 IC50 = 379 nM T87554 CM12OQ 53475998 Ki = 130 nM T87554 C6W0PN 53476000 Ki = 2100 nM T87554 C4G2ST 53476104 Ki = 95 nM T87554 C37PHN 53497571 IC50 = 3940 nM T87554 CCF1B3 53497572 IC50 = 1 nM T87554 COF6B0 54577892 IC50 = 0.17 nM T87554 C2ECL9 54577896 IC50 = 1.6 nM T87554 CY5C8A 54589404 IC50 = 0.8 nM T87554 CS7E0A 54672927 IC50 = 106.2 nM T87554 CHZ27O 54673255 IC50 = 22.4 nM T87554 C7X5ZM 54673258 IC50 = 44.3 nM T87554 CZ84NW 54673259 IC50 = 10.8 nM T87554 CX0U2A 54673422 IC50 = 32.6 nM T87554 C19FZK 54673425 IC50 = 355.2 nM T87554 CBPT15 54673763 IC50 = 1010 nM T87554 C36BAI 54673911 IC50 = 10.9 nM T87554 CD8ZK6 54674056 IC50 = 70 nM T87554 CFTE97 54674369 IC50 = 250 nM T87554 CUCI05 54674990 IC50 = 43 nM T87554 CH0IM9 54754557 IC50 = 0.7 nM T87554 C1ZF5H 54754832 Ki > 3200 nM T87554 CY9KA8 54755181 Ki > 3200 nM T87554 CE1ZK6 54759168 IC50 > 10000 nM T87554 C1XS2J 54760383 IC50 = 1200 nM T87554 CXH2P4 54766274 IC50 = 74 nM T87554 CD28VZ 54766423 IC50 = 100 nM T87554 CAP1J7 54766425 IC50 = 340 nM T87554 C75JFM 54766426 IC50 = 800 nM T87554 CDIC43 54766427 IC50 = 77 nM T87554 C2XDG1 54766428 IC50 = 380 nM T87554 C0XCY1 54766576 IC50 = 75 nM T87554 CPH3Y7 54766578 IC50 = 190 nM T87554 C0T4SL 54766726 IC50 = 83 nM T87554 CZD70Q 54767039 IC50 = 4.8 nM T87554 CN1DZ6 54767189 IC50 = 5.4 nM T87554 C83VCG 56587966 IC50 = 91 nM T87554 C1W3EZ 56591424 IC50 = 0.6 nM T87554 CTB63S 56591428 IC50 = 13 nM T87554 CWR1P6 56591446 IC50 = 0.8 nM T87554 C6ZL7H 56592816 IC50 = 81 nM T87554 C6Z1QA 56592817 IC50 = 1.2 nM T87554 C9IY4P 56594654 IC50 = 100 nM T87554 CG4E7C 56594655 IC50 = 19 nM T87554 C21GRJ 56594656 IC50 = 2700 nM T87554 CD7FW6 56594657 IC50 = 59 nM T87554 C67KYZ 56594658 IC50 = 23 nM T87554 CN96IU 56594659 IC50 = 110 nM T87554 CWYN98 56594660 IC50 = 70 nM T87554 CVDL32 56594786 IC50 = 180 nM T87554 CSE7W1 56594788 IC50 = 13 nM T87554 C0FCD9 56594790 IC50 = 23 nM T87554 CKZ27O 56594916 IC50 = 9 nM T87554 CR70XD 56595052 IC50 = 3 nM T87554 C3DJO1 56595053 IC50 = 12 nM T87554 C8KO5T 56595054 IC50 = 4 nM T87554 CW4QC9 56595056 IC50 = 8 nM T87554 C5KR6N 56595558 Ki = 67 nM T87554 COI9U2 56595687 Ki > 4000 nM T87554 C2AM6B 56595688 Ki > 4000 nM T87554 CFY2I4 56595689 Ki > 4000 nM T87554 CAM8E1 56595690 Ki = 590 nM T87554 CN5EV7 56595691 Ki > 4000 nM T87554 C6ET0W 56595693 Ki > 4000 nM T87554 CM8JX1 56604907 IC50 = 1000 nM T87554 CTR10F 56658543 Ki > 4000 nM T87554 C9HQ6G 56659204 IC50 = 12 nM T87554 C1FA3D 56659205 IC50 = 1100 nM T87554 C2E7VD 56666167 IC50 = 12 nM T87554 CGF4J3 56666168 IC50 = 14 nM T87554 CEH31Y 56668417 IC50 = 0.2 nM T87554 CG3Z0E 56669566 IC50 = 10 nM T87554 CC73NZ 56676392 IC50 = 5 nM T87554 CR23VJ 56679727 IC50 = 13 nM T87554 CXF9T4 56679728 IC50 = 41 nM T87554 CY1QA2 56683053 IC50 = 370 nM T87554 CR9A5O 56834874 IC50 = 2400 nM T87554 C58MSV 56834889 IC50 = 1620 nM T87554 CUT2G8 56835062 IC50 = 2.5 nM T87554 CJBL48 56925034 IC50 = 50 nM T87554 CBFR12 56925356 IC50 = 48 nM T87554 C80DRA 56925357 IC50 = 72 nM T87554 C0HUN8 56925358 IC50 = 100 nM T87554 C6Z2EA 56925359 IC50 = 1170 nM T87554 CC1MN2 56925454 IC50 = 1170 nM T87554 C3XC0T 56925455 IC50 = 27 nM T87554 CBW6T3 56925456 IC50 = 10 nM T87554 C8G3NO 56925457 IC50 = 2890 nM T87554 CHS19C 56925458 IC50 = 1370 nM T87554 CBMO42 56925459 IC50 = 8 nM T87554 CQTD41 56925550 IC50 = 135 nM T87554 CI9T3S 56925551 IC50 = 5 nM T87554 CS84ZU 56925552 IC50 = 4720 nM T87554 C9IVD0 56929216 Ki = 12 nM T87554 C0BO4X 56934550 Ki = 62 nM T87554 C5FY9U 56945728 IC50 = 250 nM T87554 C7D0EY 56946378 IC50 = 1700 nM T87554 CUQ50W 56946379 IC50 = 18 nM T87554 C3B2YH 56951311 IC50 = 0.17 nM T87554 CJMB49 56953110 Ki = 26 nM T87554 CAK91L 56955954 IC50 > 3600 nM T87554 CSO40C 56973425 Ki = 4.4 nM T87554 CU5BD9 57336812 IC50 = 1.8 nM T87554 C31LJU 57339437 Ki = 200 nM T87554 CMF7J0 57339438 Ki = 250 nM T87554 CPO2J4 57342178 IC50 = 150 nM T87554 C72PED 57342179 IC50 = 63 nM T87554 CA93PN 57342180 IC50 = 370 nM T87554 CI70CT 57345538 IC50 = 650 nM T87554 CVS76D 57390492 IC50 = 0.5 nM T87554 C4P5YQ 57390669 IC50 = 0.54 nM T87554 C3N2SF 57390670 IC50 = 1.1 nM T87554 COV39R 57390671 IC50 = 0.5 nM T87554 C9MW1O 57390672 IC50 = 0.3 nM T87554 CBJ93Q 57390673 IC50 = 0.4 nM T87554 C10WYL 57390861 IC50 = 16 nM T87554 CC7LW5 57392473 IC50 = 0.23 nM T87554 CEDR08 57392474 IC50 = 1 nM T87554 C79QPH 57392475 IC50 = 0.5 nM T87554 CS2R7J 57392476 IC50 = 0.36 nM T87554 C5O1HP 57392676 IC50 = 2.1 nM T87554 C6SKR3 57392677 IC50 = 6.3 nM T87554 C16RBI 57393424 IC50 = 450 nM T87554 C56DZN 57394024 IC50 = 0.6 nM T87554 C93GNJ 57394178 IC50 = 0.33 nM T87554 CZI79U 57394179 IC50 = 1.2 nM T87554 C0ZSA5 57394180 IC50 = 0.4 nM T87554 C3J4NV 57394381 IC50 = 2 nM T87554 CK74ND 57394382 IC50 = 0.22 nM T87554 C43EQN 57394383 IC50 = 0.52 nM T87554 C1V9MC 57394384 IC50 = 16 nM T87554 CKS67A 57396146 IC50 = 0.22 nM T87554 CE4FA1 57396924 IC50 = 330 nM T87554 CWJ70D 57397964 IC50 = 62 nM T87554 CAQ9D6 57397965 IC50 = 2900 nM T87554 CE8JW3 57398441 IC50 = 1.5 nM T87554 CFU5H3 57399413 IC50 = 2.1 nM T87554 C8CTY7 57399414 IC50 = 0.47 nM T87554 CKE7L0 57399415 IC50 = 0.35 nM T87554 C8BD2Q 57399416 IC50 = 480 nM T87554 CZX8R7 57399606 IC50 = 0.09 nM T87554 CMU89A 57401172 IC50 = 3.7 nM T87554 C43NFS 57401173 IC50 = 1 nM T87554 CL9Z2D 57401363 IC50 = 0.64 nM T87554 C8F4ME 57401364 IC50 = 0.27 nM T87554 CZTG84 57402768 IC50 = 0.9 nM T87554 CK06MA 57402935 IC50 = 1.14 nM T87554 CZ85FM 57402936 IC50 = 0.5 nM T87554 C9WMS3 57402937 IC50 = 0.8 nM T87554 C0FS4C 57402938 IC50 = 0.35 nM T87554 C9GN1M 57403118 IC50 = 0.6 nM T87554 C56CSP 57403119 IC50 = 39 nM T87554 C6A8WC 57502370 IC50 = 2132 nM T87554 CIO15D 57502371 IC50 > 10000 nM T87554 C6YOU9 57502372 IC50 = 1406 nM T87554 C8DN1A 57502373 IC50 = 2874 nM T87554 C15XOS 57502374 IC50 = 2165 nM T87554 CEF53Z 57502376 IC50 = 47 nM T87554 CTY54N 57502377 IC50 = 136 nM T87554 CBLN61 57502378 IC50 = 8 nM T87554 CDV4R1 57502379 IC50 = 1.5 nM T87554 CILJ54 57502380 IC50 = 1615 nM T87554 CS90RX 57502381 IC50 = 3 nM T87554 CE6B7C 57502382 IC50 = 0.8 nM T87554 CC82QJ 57502383 IC50 = 3.1 nM T87554 C72OWZ 57502386 IC50 = 1.1 nM T87554 CHC90Q 57502387 IC50 = 1.4 nM T87554 C9Z6QJ 57502388 IC50 = 0.7 nM T87554 CMF31G 57502390 IC50 = 26 nM T87554 C4QXU9 57514090 IC50 = 193 nM T87554 C0YW2D 57514091 IC50 = 5.6 nM T87554 CU8Y3P 57514092 IC50 = 1.3 nM T87554 C5K3VZ 57514093 IC50 = 4 nM T87554 CNQ6K8 57659282 IC50 = 617 nM T87554 CS75LF 57659335 IC50 = 20 nM T87554 COU4M1 57915982 IC50 = 17 nM T87554 C1G5SK 57916044 IC50 = 23 nM T87554 C3C0PQ 57916049 IC50 = 43 nM T87554 CH6RB0 57916164 IC50 = 23 nM T87554 C9MF8U 57928260 IC50 = 11 nM T87554 C3KQJ8 57928435 IC50 = 1.7 nM T87554 C5H8VE 57928583 IC50 = 11 nM T87554 C13VIO 57928632 IC50 = 120 nM T87554 C8BTO7 57928826 IC50 = 5 nM T87554 C18MVX 57990771 IC50 = 5000 nM T87554 C4TQ9L 57990797 IC50 = 5.7 nM T87554 C4XC3V 57990957 IC50 > 980 nM T87554 CB6F5S 57990969 IC50 = 0.9 nM T87554 C13BGJ 57991037 IC50 = 7.9 nM T87554 CDRB84 57991074 IC50 = 129.9 nM T87554 CJ4B2L 57991089 IC50 = 621.7 nM T87554 C9EA1S 57991186 IC50 = 1431.3 nM T87554 C5B3HI 57991212 IC50 = 2.9 nM T87554 C48LZT 57991260 IC50 > 980 nM T87554 C8R4FE 57991377 IC50 = 2.2 nM T87554 C19UKS 57991389 IC50 = 5.2 nM T87554 C1KH5D 57991398 IC50 = 1.7 nM T87554 CSN47V 57991473 IC50 = 8.7 nM T87554 CD6ZP3 58009815 EC50 = 1600 nM T87554 CWU1Y3 58009825 EC50 = 890 nM T87554 C8S6MY 58010054 EC50 = 4200 nM T87554 CM1B4V 58010265 EC50 = 4800 nM T87554 CGR87Y 58063067 Ki = 1.3 nM T87554 C3J7XM 58063084 Ki = 1 nM T87554 CW2Z5I 58063100 Ki = 0.3 nM T87554 C1EVX0 58063117 Ki = 0.1 nM T87554 C7NE0H 58063121 Ki = 0.1 nM T87554 COT5L0 58063146 Ki = 1.6 nM T87554 CGBY54 58063225 Ki = 1 nM T87554 C1RF4W 58063241 Ki = 31.9 nM T87554 C0P8VW 58063334 Ki = 2.5 nM T87554 CZO2J1 58063487 Ki = 5.1 nM T87554 C2U5TY 58063491 Ki = 1.8 nM T87554 CQND09 58177229 IC50 = 102 nM T87554 CU4I8X 58177247 IC50 = 71 nM T87554 CLEH36 58177279 IC50 = 54 nM T87554 CIK3U8 58177332 IC50 = 36 nM T87554 C8D2TA 58177362 IC50 = 181 nM T87554 CYC85B 58177456 IC50 = 9 nM T87554 C7BU0H 58180518 IC50 = 3.1 nM T87554 CKA28H 58180521 IC50 = 1.2 nM T87554 C2I5LO 58180525 IC50 = 2.1 nM T87554 CN4OZ8 58180573 IC50 = 1.4 nM T87554 C92FOB 58180591 IC50 = 0.9 nM T87554 CWXC70 58180596 IC50 = 2.5 nM T87554 C9N1QB 58180623 IC50 = 1.5 nM T87554 CSK1U8 58180628 IC50 = 1.4 nM T87554 C6LT9S 58180630 IC50 = 1.9 nM T87554 CCBT87 58180639 IC50 = 1.4 nM T87554 C7Q8YZ 58374808 IC50 > 10000 nM T87554 CP81TW 58394456 Ki = 59 nM T87554 C4H3FY 58394522 Ki = 20 nM T87554 CM6SK2 58394565 Ki = 32 nM T87554 C6HPO3 58394632 Ki = 15 nM T87554 CK71MA 58394722 Ki = 580 nM T87554 CO5TH6 58394820 Ki = 47 nM T87554 CY0UV6 58394828 Ki = 2.9 nM T87554 CW7D0O 58394866 Ki = 21 nM T87554 C0W2AT 58394878 Ki = 669 nM T87554 C97QAK 58394904 Ki = 18 nM T87554 C9Q4WD 58394916 Ki = 25 nM T87554 CI37CQ 58394927 Ki = 5 nM T87554 C5RGU7 58394946 Ki = 721 nM T87554 C6KO0G 58395044 IC50 = 5700 nM T87554 CDK5L1 58395223 Ki = 3.8 nM T87554 C9J5UV 58395232 Ki = 11 nM T87554 CYC87B 58395253 Ki = 487 nM T87554 C5S8BK 58395290 Ki = 66 nM T87554 C4H2ZP 58395301 Ki = 8.3 nM T87554 C28ADB 58395446 Ki = 2.1 nM T87554 CLA5V3 58395468 Ki = 121 nM T87554 C0X5CV 58395476 Ki = 3.7 nM T87554 C9TV2G 58398904 IC50 = 490 nM T87554 CR9T7W 58438557 IC50 = 2030 nM T87554 CY3W6B 58438580 IC50 = 134.2 nM T87554 CR7C4V 58438607 IC50 = 0.8 nM T87554 C9MIL7 58450666 IC50 = 203 nM T87554 CWX4G9 58522116 IC50 = 2320 nM T87554 C4A6LT 58522124 IC50 = 1710 nM T87554 CI9VB0 58522237 IC50 = 580 nM T87554 C1LE9A 58522238 IC50 = 900 nM T87554 C74ACR 58522276 IC50 = 1000 nM T87554 CI0L1J 58522322 IC50 = 1210 nM T87554 CVMO97 58522377 IC50 = 1250 nM T87554 C7S1PR 58522381 IC50 = 410 nM T87554 C2W0OD 58539094 Ki > 3200 nM T87554 C6CDB7 58539140 Ki = 3000 nM T87554 CB3TQ8 58539146 Ki > 3200 nM T87554 C7WRQ5 58539268 Ki > 3200 nM T87554 C97ZGJ 58539301 Ki > 3200 nM T87554 C8X6YE 58557497 IC50 = 11400 nM T87554 CX0Q2W 58688109 IC50 = 804 nM T87554 C6BPR2 58985201 IC50 > 30000 nM T87554 C3YHW8 59186181 Ki = 5 nM T87554 C5MHP0 59186191 Ki = 4.8 nM T87554 CSR49F 59186194 Ki = 17.7 nM T87554 CT8CI4 59186216 Ki = 19.3 nM T87554 CGS2D4 59186263 Ki = 3 nM T87554 CHG45P 59186268 Ki = 0.6 nM T87554 C8NA2Z 59186270 Ki = 40.6 nM T87554 C2AF7G 59186271 Ki = 70.9 nM T87554 CI93GZ 59186442 Ki = 9.1 nM T87554 C4XQ9E 59186482 Ki = 2 nM T87554 CS07KJ 59186487 Ki = 0.9 nM T87554 CD30LA 59186489 Ki = 0.3 nM T87554 CGRE28 59198979 Ki = 0.5 nM T87554 CG4Y8K 59198994 Ki = 0.5 nM T87554 C4TJS9 59199010 Ki = 0.4 nM T87554 CPD28H 59199061 Ki = 1.4 nM T87554 CJA50L 59199121 Ki = 0.7 nM T87554 C3S1CI 59199131 Ki = 0.6 nM T87554 CR6UM8 59199136 Ki = 1.1 nM T87554 CR2OB1 59199142 Ki = 0.6 nM T87554 C6TAW4 59199165 Ki = 0.5 nM T87554 CPWM60 59291925 IC50 = 12 nM T87554 C3CV0R 59291929 IC50 = 46 nM T87554 COXI75 59291940 IC50 = 370 nM T87554 CE6KO4 59291951 IC50 = 17 nM T87554 CT3EW2 59292007 IC50 = 3.2 nM T87554 C2PE0T 59292008 IC50 = 41 nM T87554 CU3W2S 59292043 IC50 = 49 nM T87554 CC6J4I 59363349 EC50 = 452 nM T87554 CQ93TM 59363383 EC50 = 778 nM T87554 CKQ31B 59363409 EC50 = 798 nM T87554 CZ3TG1 59375154 IC50 = 212 nM T87554 CU7Q5A 59435986 IC50 = 2 nM T87554 C64IHJ 59435987 IC50 = 7 nM T87554 C2VG8U 59436001 IC50 = 1 nM T87554 CCJ81A 59436022 IC50 = 37 nM T87554 CG9NO0 59436049 IC50 = 0.9 nM T87554 CT4P2H 59436062 IC50 = 0.8 nM T87554 C7T9PR 59436066 IC50 = 0.15 nM T87554 C8D5BA 59436080 IC50 = 9 nM T87554 CRV24D 59436099 IC50 = 3 nM T87554 CP9BH2 59436109 IC50 = 0.5 nM T87554 C81AOP 59525628 IC50 = 178 nM T87554 CI0G2S 59525684 IC50 = 93 nM T87554 C3R7ZX 59525688 IC50 = 140 nM T87554 CP3SN6 59525717 IC50 = 36 nM T87554 CT35BZ 59525728 IC50 = 690 nM T87554 CVD4E5 59525760 IC50 = 80 nM T87554 CP1F6X 59526007 IC50 = 380 nM T87554 CM7OV6 59526068 IC50 = 155 nM T87554 C4N9MS 59526260 IC50 = 312 nM T87554 CFEU09 59589639 Ki = 207 nM T87554 C0DV7R 59589757 Ki = 59 nM T87554 CMPO72 59599420 IC50 = 215 nM T87554 CXJ63M 59603829 IC50 = 1200 nM T87554 CQEU96 59603842 IC50 = 64 nM T87554 CDMO01 59617921 Ki > 3500 nM T87554 CUNY05 59617942 Ki > 3500 nM T87554 CY7V3I 59617971 Ki = 1400 nM T87554 CM6B3E 59618010 Ki = 380 nM T87554 CQCG48 59618036 Ki = 2500 nM T87554 CJ5GF1 59618081 Ki > 3500 nM T87554 CT12JO 59618117 Ki = 860 nM T87554 C42OZL 59618123 Ki = 55 nM T87554 COI26N 59618146 Ki > 3500 nM T87554 CR5GJ4 59618147 Ki = 1300 nM T87554 C9GB1C 59618160 Ki = 2400 nM T87554 CR9F7D 59618164 Ki = 310 nM T87554 C7XWE2 59618171 Ki = 510 nM T87554 C2EIA3 59618285 Ki = 130 nM T87554 C1ZKR9 59618313 Ki = 2900 nM T87554 C26BNV 59618424 Ki = 2700 nM T87554 C3B7CU 59618428 Ki = 63 nM T87554 CBH83T 59618445 Ki = 60 nM T87554 C3HC4P 59618462 Ki = 2400 nM T87554 CX0FQ2 59618505 Ki = 20 nM T87554 CG8ET4 59618513 Ki = 250 nM T87554 CR27IT 59618564 Ki > 3500 nM T87554 CSZA16 60155724 IC50 > 3600 nM T87554 CNY59P 60165955 Ki = 0.3 nM T87554 CY3QT8 60165956 Ki = 25 nM T87554 CKT4Y7 60170769 Ki = 6.4 nM T87554 C3YSV5 60170770 Ki = 74 nM T87554 C34RVN 60170771 Ki = 9.3 nM T87554 C74FPI 60170772 Ki = 11 nM T87554 CTC8E4 60170773 Ki = 17 nM T87554 CR80CH 60170858 Ki = 12 nM T87554 C3PA9G 60170859 Ki = 21 nM T87554 C2AEG3 60170860 Ki = 520 nM T87554 CHJM71 60170861 Ki = 26 nM T87554 CBP48G 60170862 Ki = 28 nM T87554 C3R0NO 63107904 IC50 = 3960 nM T87554 CK6WO0 66552478 IC50 < 10000 nM T87554 CE4RV7 66558256 IC50 > 10000 nM T87554 CQK4Y2 66570958 IC50 = 8 nM T87554 C5RAC8 66571005 IC50 = 12 nM T87554 CVXT19 66571006 IC50 = 308 nM T87554 C5UFY3 66571008 IC50 = 3 nM T87554 CG8AP3 66571009 IC50 = 187 nM T87554 C20EXP 66571075 IC50 = 24 nM T87554 C3WF4H 66571076 IC50 = 10 nM T87554 C3IRH5 66571077 IC50 = 150 nM T87554 CYS96O 66571078 IC50 = 21 nM T87554 CPW01U 66571135 IC50 = 2 nM T87554 C32BMH 66571136 IC50 = 53 nM T87554 CC04XH 66571138 IC50 = 35 nM T87554 CI6A2Z 66571139 IC50 = 109 nM T87554 CGP12A 66571140 IC50 = 57 nM T87554 CJL68E 66571195 IC50 = 46 nM T87554 C6STC7 66571196 IC50 = 247 nM T87554 C3U6ED 66571199 IC50 = 268 nM T87554 CQ49JM 66571200 IC50 = 114 nM T87554 CY3P8G 66571201 IC50 = 3056 nM T87554 CYFL93 66571254 IC50 = 44 nM T87554 C5H1VS 66571255 IC50 = 154 nM T87554 CG3XE8 66571256 IC50 = 384 nM T87554 C3WM6R 66571316 IC50 = 43 nM T87554 C8DSK2 66571317 IC50 = 1235 nM T87554 C72WVF 66571377 IC50 = 66 nM T87554 C9T4VJ 66571378 IC50 = 1537 nM T87554 CJ08ZL 66604045 IC50 = 5.7 nM T87554 CY0I2V 66604274 IC50 = 370 nM T87554 CD0LJ6 66604359 IC50 = 2.4 nM T87554 CS8HK2 66604394 IC50 = 120 nM T87554 C7U8GC 66604464 IC50 = 110 nM T87554 CXU94O 66604576 IC50 = 17 nM T87554 CE9T0V 66604664 IC50 = 86 nM T87554 C7WO4A 66604791 IC50 = 3.1 nM T87554 CW53KR 66604810 IC50 = 130 nM T87554 CNW05G 66604855 IC50 = 6.8 nM T87554 CT4RU2 66604890 IC50 = 1.7 nM T87554 C0JS8O 66604914 IC50 = 1.2 nM T87554 CW9LD1 66604921 IC50 = 8 nM T87554 CTMX20 66605009 IC50 = 7.4 nM T87554 C0EVU7 66605043 IC50 = 27 nM T87554 CP0DB1 66605115 IC50 = 10.2 nM T87554 CGS8J2 66605151 IC50 = 4.3 nM T87554 CB1WC9 66605298 IC50 = 3.5 nM T87554 CCWU74 66605322 IC50 = 16 nM T87554 C7Q8ZG 66605359 IC50 = 7.4 nM T87554 C16TEK 66605475 IC50 = 6.1 nM T87554 C7MOJ6 66605487 IC50 = 470 nM T87554 CDZA70 66605639 IC50 = 5.2 nM T87554 C53NBQ 66605756 IC50 = 280 nM T87554 CN5BR8 66605844 IC50 = 2.6 nM T87554 CDES25 66606401 IC50 = 6.2 nM T87554 C5J4MR 66850717 Ki = 3.2 nM T87554 CC6JF4 66851197 Ki = 3.2 nM T87554 CO2H4Q 66851201 Ki = 49 nM T87554 C3BTX2 66851307 Ki = 41.2 nM T87554 C7ONK1 66851426 Ki = 2.1 nM T87554 C5PVB2 67008690 IC50 = 194 nM T87554 C8OZ6W 67008828 IC50 = 84 nM T87554 C1HSE0 67035086 IC50 = 1100 nM T87554 CWI6K5 67035106 IC50 > 10000 nM T87554 C38RGB 67035556 IC50 > 10000 nM T87554 CZX1E0 67123420 IC50 = 68 nM T87554 C0RCI2 67123577 IC50 = 0.3 nM T87554 C37NKO 67129970 IC50 = 4920 nM T87554 CK80LJ 67130050 IC50 = 4170 nM T87554 CV63UL 67240318 IC50 > 10000 nM T87554 C6YHJ5 67277266 IC50 = 430 nM T87554 C78TXA 67277273 IC50 = 200 nM T87554 C0O7TC 67277276 IC50 = 2.6 nM T87554 C3YK7Q 67277763 IC50 = 310 nM T87554 CQXW93 67277840 IC50 = 850 nM T87554 CF4AB0 67277979 IC50 = 1800 nM T87554 CFM39N 67278030 IC50 = 640 nM T87554 C5U2IW 67278045 IC50 = 23 nM T87554 CS9K0L 67278047 IC50 = 140 nM T87554 C2FW8H 67278142 IC50 = 85 nM T87554 CQRS42 67278151 IC50 = 82 nM T87554 C5V9DZ 67278165 IC50 = 500 nM T87554 CMJ29W 67278195 IC50 = 88 nM T87554 C2C7BD 67278380 IC50 = 190 nM T87554 CVL35U 67278385 IC50 = 97 nM T87554 CKVB79 67278425 IC50 = 17 nM T87554 C2C1RE 67329237 IC50 > 30000 nM T87554 CV80IQ 67330694 IC50 = 27 nM T87554 C16THB 67351896 Ki = 27 nM T87554 CFX84K 67352945 Ki = 21 nM T87554 C1FLT6 67354280 Ki = 401 nM T87554 CEF67O 67383086 Ki = 14 nM T87554 CLO13H 67383145 Ki = 110 nM T87554 C94UAF 67383148 Ki = 43 nM T87554 C5D2QA 67383227 Ki = 93 nM T87554 C4AE8Z 67383253 Ki = 10 nM T87554 CW8Q3F 67383552 Ki = 5.4 nM T87554 C6UF3T 67383612 Ki = 21 nM T87554 CV38SD 67383669 Ki = 440 nM T87554 C9WY2P 67383875 Ki = 22 nM T87554 CJ2Q1S 67383893 Ki = 26 nM T87554 CUK87J 67387753 Ki = 150 nM T87554 C14RKJ 67479440 IC50 > 100000 nM T87554 C5WQC2 67502257 IC50 > 1000 nM T87554 CZ0O6N 68234726 Ki = 16 nM T87554 CA89HR 68235185 Ki = 490 nM T87554 CYR38C 68241014 IC50 = 400 nM T87554 C0MY1I 68241371 IC50 = 130 nM T87554 CX6S4E 68254533 IC50 = 800 nM T87554 C4U1IR 68291322 IC50 = 42 nM T87554 C2P7DB 68291391 IC50 = 280 nM T87554 CRM3S0 68291627 IC50 = 210 nM T87554 C4LKB3 68291752 IC50 = 18 nM T87554 CQ49HB 68291755 IC50 = 70 nM T87554 CXI4L1 68291797 IC50 = 170 nM T87554 C8T5VB 68291830 IC50 = 62 nM T87554 CPRW18 68291866 IC50 = 438 nM T87554 C6UWI3 68291981 IC50 = 130 nM T87554 CYN89R 68292156 IC50 = 120 nM T87554 C76EZC 68292170 IC50 = 130 nM T87554 CGA0W6 68292183 IC50 = 31 nM T87554 C93LZT 68292196 IC50 = 130 nM T87554 C8I7GC 68293638 IC50 > 10000 nM T87554 CD56XK 68293660 IC50 > 10000 nM T87554 CYI75G 68678653 IC50 > 30000 nM T87554 C7GRV2 68755406 IC50 = 2320 nM T87554 CIL58T 69023801 IC50 = 12.8 nM T87554 C5DGR9 69036886 IC50 = 1173 nM T87554 CK8DC3 69046862 IC50 = 15 nM T87554 CV0K3P 69267827 IC50 = 4 nM T87554 CVH5M3 69671224 Ki = 190 nM T87554 COX56A 69809432 IC50 = 45 nM T87554 CECG39 69809726 IC50 = 108 nM T87554 C7FA5L 69811602 EC50 = 3690 nM T87554 C92EAC 69811936 EC50 = 2665 nM T87554 C0XO1M 69812740 IC50 = 82 nM T87554 CJ96RN 70099013 Ki > 3200 nM T87554 CRZ5V2 70495652 Ki = 63.3 nM T87554 CS47OP 70496411 Ki = 11.9 nM T87554 CV0NP6 70496595 Ki = 0.4 nM T87554 CK5H1Y 70497007 Ki = 103 nM T87554 CTG78Y 70497097 Ki = 5.6 nM T87554 CTY17Z 70497535 Ki = 16.7 nM T87554 C6NSG3 70497750 Ki = 9.7 nM T87554 CWP52K 70497865 Ki = 15.5 nM T87554 CP48DJ 70498203 Ki = 41.1 nM T87554 CQH47T 70498861 Ki = 14 nM T87554 C7VJ6A 70647728 IC50 = 370 nM T87554 CASQ98 70650259 IC50 = 90 nM T87554 CQ2F8J 70824464 Ki = 610 nM T87554 CBF3Q6 71042865 IC50 = 972 nM T87554 CNR2Y9 71061323 IC50 = 1.3 nM T87554 C51JTW 71061588 IC50 = 1.7 nM T87554 CF69WT 71061828 IC50 = 3.6 nM T87554 COU2C5 71061858 IC50 = 7.4 nM T87554 CW9OE6 71061878 IC50 = 2 nM T87554 CK9LZ3 71061981 IC50 = 1.9 nM T87554 CU1T4P 71061987 IC50 = 5.3 nM T87554 CJH94D 71062030 IC50 = 1.5 nM T87554 CUW46K 71062043 IC50 = 4.3 nM T87554 C05VNE 71062076 IC50 = 4.8 nM T87554 C4AC9U 71212257 IC50 < 0.2 nM T87554 COD6B2 71222450 Ki = 34 nM T87554 COR71Z 71285696 IC50 = 740 nM T87554 C3ZL5S 71285760 IC50 = 56 nM T87554 CME92O 71285933 IC50 = 15 nM T87554 C2FL6H 71286084 IC50 = 1.3 nM T87554 C14YOJ 71286184 IC50 = 13 nM T87554 CX23BP 71288497 IC50 = 20 nM T87554 CH1AJ3 71288512 IC50 = 1.1 nM T87554 CA1T5H 71288539 IC50 = 16 nM T87554 CYU2Z4 71288594 IC50 = 28 nM T87554 CBY4K0 71288602 IC50 = 22 nM T87554 CWLC45 71288607 IC50 = 38 nM T87554 CDST08 71288618 IC50 = 10800 nM T87554 C45HTF 71288693 IC50 = 3.3 nM T87554 COC20B 71288707 IC50 = 83 nM T87554 C6JD3S 71288724 IC50 = 4.2 nM T87554 COV78A 71288729 IC50 = 5.9 nM T87554 C8DY1N 71288732 IC50 = 57 nM T87554 CNV7B6 71300296 Ki = 0.72 nM T87554 C49STX 71450071 Ki = 5.2 nM T87554 CX4LE5 71453548 Ki = 7 nM T87554 CPO7Y1 71454973 Ki = 12 nM T87554 CAN57Z 71455263 Ki > 3200 nM T87554 CKT60L 71455860 Ki = 920 nM T87554 C4D1TQ 71456076 IC50 > 980 nM T87554 CPY5K3 71457046 Ki > 3200 nM T87554 C1X6YV 71457047 Ki = 3 nM T87554 CML7F1 71458913 Ki = 64 nM T87554 CFN35P 71459077 Ki = 0.6 nM T87554 CR6O7Q 71462440 Ki > 3200 nM T87554 C01XHF 71510730 IC50 = 392 nM T87554 C09YSR 71510731 IC50 = 594 nM T87554 C9DIK2 71512060 IC50 > 10000 nM T87554 CCN01X 71547862 IC50 > 10000 nM T87554 CVEO06 71558636 IC50 = 39 nM T87554 C07SFW 71600166 IC50 = 1350 nM T87554 CWJ1G4 71600167 IC50 = 446 nM T87554 CKY79O 71615499 Ki = 1.41 nM T87554 C8GLY0 71615500 IC50 = 4 nM T87554 CA7Q3S 71615501 IC50 = 3 nM T87554 CVYS15 71617859 IC50 = 3.2 nM T87554 C7T5LI 71655637 Ki = 1232 nM T87554 CT3M4B 71655638 Ki = 446 nM T87554 CSC81X 71655639 Ki = 57 nM T87554 C3U1ZV 71655709 Ki = 17 nM T87554 CE1JQ3 71655774 Ki = 33 nM T87554 CX5OU4 71681533 Ki = 18 nM T87554 C29FVT 71681534 Ki = 90 nM T87554 C7WQP2 71681535 Ki = 76 nM T87554 CEQM71 71681536 EC50 > 10 nM T87554 CV5FB0 71681691 Ki = 44 nM T87554 C6JH7K 71681692 Ki = 49 nM T87554 CS62NH 71698376 IC50 = 111900 nM T87554 CI8X1R 71698379 IC50 = 138200 nM T87554 C5QK6S 71727668 IC50 = 26 nM T87554 C8PSM2 71737832 Ki = 145 nM T87554 CO76WG 71818715 Ki = 8 nM T87554 CR02FG 71818862 Ki = 2200 nM T87554 CY6WE7 71818863 Ki = 2200 nM T87554 CW52BU 71943288 IC50 = 2380 nM T87554 C54XWG 72190869 IC50 > 10000 nM T87554 C4XY6C 72195599 IC50 = 126 nM T87554 CLD12K 72201823 IC50 = 2.7 nM T87554 CYQN46 72201826 IC50 = 4.1 nM T87554 CP9CJ3 72201957 IC50 = 164 nM T87554 CMVI93 72201958 IC50 = 37.9 nM T87554 CD9Z4H 72202092 IC50 = 3.7 nM T87554 CLIS85 72202093 IC50 = 9.4 nM T87554 C5Q7YT 72202095 IC50 = 12.1 nM T87554 C8NGE4 72202097 IC50 = 42.9 nM T87554 C1W6LK 72202246 IC50 = 55.4 nM T87554 C6W4ZS 72202247 IC50 = 4.2 nM T87554 C1N7LQ 72202249 IC50 = 0.5 nM T87554 C2W6TI 72202397 IC50 = 1.6 nM T87554 CIKL36 72202398 IC50 = 9.6 nM T87554 C1I4LX 72202399 IC50 = 3125 nM T87554 C4CB2S 72202400 IC50 = 53.7 nM T87554 CVI63X 72202547 IC50 = 1.6 nM T87554 C0EZ3I 72202548 IC50 = 2.9 nM T87554 C7OY3V 72202549 IC50 = 14.2 nM T87554 CH40KC 72202550 IC50 = 9.2 nM T87554 CA5CI3 72202825 IC50 = 6.4 nM T87554 C6THF4 72374600 Ki = 70 nM T87554 CHK46S 72375658 Ki = 123 nM T87554 COPS30 72375659 Ki = 377 nM T87554 CB9ZL4 72375660 Ki = 130 nM T87554 C0K5IO 72375661 Ki = 54 nM T87554 C7PG8Z 72375662 Ki = 189 nM T87554 CCZO42 72375759 Ki = 550 nM T87554 CEV9X5 72375760 Ki = 201 nM T87554 COE6R4 72375761 Ki = 766 nM T87554 C1G8RD 72375763 Ki = 690 nM T87554 C8SLE9 72375764 Ki = 380 nM T87554 C74WLS 72375765 Ki = 3200 nM T87554 CP2KL5 72375766 Ki = 3200 nM T87554 CT9D3J 72375844 Ki = 1500 nM T87554 CZN81X 72375845 Ki = 567 nM T87554 CXL52K 72375846 Ki = 1400 nM T87554 CAV52F 72375847 Ki = 575 nM T87554 C3QT2E 72375850 Ki = 63 nM T87554 C0UJ9M 72375852 Ki = 150 nM T87554 CNJ03L 72375990 Ki > 3500 nM T87554 C5R0WV 72375991 Ki = 3200 nM T87554 CVUL48 72375992 Ki = 1800 nM T87554 CO8KW2 72375993 Ki > 3500 nM T87554 CN0I2W 72375994 Ki > 3500 nM T87554 C1XD7U 72375995 Ki = 3100 nM T87554 C8BJ4U 72375996 Ki > 3500 nM T87554 C7XFW2 72375997 Ki > 3500 nM T87554 CJB95D 72375998 Ki > 3500 nM T87554 CS5V9L 72376089 Ki = 1400 nM T87554 C37GPL 72376090 Ki = 2000 nM T87554 C9U3WO 72376091 Ki > 3500 nM T87554 C0DL3F 72698602 IC50 < 1 nM T87554 CK7F6U 72700776 Ki = 1 nM T87554 CLOE10 72706962 IC50 = 575 nM T87554 C1D2AM 72737634 IC50 = 1 nM T87554 CG16YE 72771106 IC50 = 460 nM T87554 CMK8Z4 73055651 IC50 = 3 nM T87554 C50CRU 73056517 IC50 = 1 nM T87554 CQAI18 73056519 IC50 = 12 nM T87554 C16AQK 73056520 IC50 = 8 nM T87554 C2ZFQ1 73057136 IC50 = 16 nM T87554 CH43OS 73057443 IC50 = 1 nM T87554 CDS4T9 73057444 IC50 = 20 nM T87554 CXD38C 73346480 Ki = 0.6 nM T87554 C0G5RD 73347974 Ki = 574 nM T87554 CRAW59 73349195 Ki = 230 nM T87554 C41ZJV 73349520 Ki = 1.8 nM T87554 CJE73Y 73352545 Ki = 23 nM T87554 CPRD59 73352546 Ki = 9 nM T87554 C4BUW7 73353407 IC50 = 20 nM T87554 CXT70E 73354035 Ki = 13 nM T87554 CGI13D 73354036 Ki = 158 nM T87554 CL4SD8 73355260 Ki > 3500 nM T87554 CMR72H 73355566 Ki = 21 nM T87554 CPT46O 73355567 Ki > 5600 nM T87554 C04CXF 73355568 Ki = 59 nM T87554 C3G2BM 73357112 Ki = 3 nM T87554 CO6F2B 73357113 Ki = 4 nM T87554 C8DSE2 75108379 IC50 < 3 nM T87554 CS41CX 75108409 IC50 = 33 nM T87554 CH20VA 75108447 IC50 = 24 nM T87554 CP90QE 75108517 IC50 < 3 nM T87554 CG6T5S 76072368 IC50 = 425.6 nM T87554 COMF95 76072369 IC50 = 10.8 nM T87554 CRK1L2 76210601 IC50 = 22 nM T87554 CO0BQ5 76310565 IC50 = 1480 nM T87554 C6ZAB2 76310566 IC50 > 10000 nM T87554 C0F6VU 76310567 IC50 > 10000 nM T87554 CDO38G 76310568 IC50 > 10000 nM T87554 CL42BQ 76310569 IC50 > 10000 nM T87554 CWI1Q4 76310570 IC50 = 1238 nM T87554 C8OY6Q 76310785 IC50 > 100000 nM T87554 CAL3U7 76310788 IC50 > 100000 nM T87554 C7SXJ1 76314208 IC50 = 1270 nM T87554 CSDI71 76314209 IC50 = 490 nM T87554 C12YAE 76314414 IC50 > 100000 nM T87554 CM6LI3 76314606 IC50 = 0.6 nM T87554 CXF1I3 76317774 IC50 > 10000 nM T87554 CY79VS 76317775 IC50 > 10000 nM T87554 CNK2I1 76317776 IC50 > 10000 nM T87554 CS02NA 76317777 IC50 = 1637 nM T87554 CAHW32 76317778 IC50 = 1270 nM T87554 CT9JM4 76317888 IC50 = 670 nM T87554 C97RBS 76317979 IC50 > 100000 nM T87554 C2SMK1 76321491 IC50 > 10000 nM T87554 C2DSX7 76321492 IC50 = 10080 nM T87554 CI2VZ6 76321886 IC50 = 26 nM T87554 CL0T7B 76322219 IC50 = 21513 nM T87554 CXA4O1 76325093 IC50 > 10000 nM T87554 CEZ64F 76325209 IC50 = 50 nM T87554 C1AI0J 76325315 IC50 > 100000 nM T87554 CPQA45 76325323 IC50 > 100000 nM T87554 C8GK0H 76328659 IC50 > 10000 nM T87554 C74RUX 76329058 IC50 = 10 nM T87554 CJN89E 76332335 IC50 > 10000 nM T87554 CW1QK4 76332336 IC50 = 2130 nM T87554 C2P1MX 76332338 IC50 = 11080 nM T87554 CB5Y0Z 76332540 IC50 > 100000 nM T87554 CB4KQ7 76335967 IC50 > 10000 nM T87554 C84PFQ 76335968 IC50 = 9687 nM T87554 CW1HQ9 76370451 IC50 = 5 nM T87554 CD6Y1F 78320046 IC50 = 550 nM T87554 CW08SU 78320048 IC50 = 220 nM T87554 CWI93D 78323836 IC50 = 381 nM T87554 C5UK9L 78323837 IC50 = 542 nM T87554 CQ3EJ1 78324132 IC50 = 6810 nM T87554 C7VOX0 78324136 IC50 = 1196 nM T87554 CA2Y8L 78324435 IC50 = 1090 nM T87554 C4I7WD 78324744 IC50 = 412 nM T87554 CQ2SU8 78673832 IC50 > 30000 nM T87554 CE0W9R 78673833 IC50 > 30000 nM T87554 CNI6U3 86267948 IC50 = 442 nM T87554 CV8UZ1 86278565 IC50 = 225 nM T87554 CZ97VP 86294733 IC50 = 680 nM T87554 CPG3A5 86302574 IC50 = 21052 nM T87554 C96EDF 86660048 IC50 = 7100 nM T87554 CC8I0M 86707711 IC50 = 15 nM T87554 CW4Z2F 89470642 IC50 = 1.2 nM T87554 CBRF87 89470690 IC50 = 2.8 nM T87554 C7B8OH 89470730 IC50 = 0.47 nM T87554 CDQ8C6 89471114 IC50 = 1.5 nM T87554 C4G5LP 89471136 IC50 = 3 nM T87554 CU6J4F 89498235 Ki = 23 nM T87554 CS7GX8 89708625 IC50 = 162400 nM T87554 C1HW4B 89735655 IC50 = 4400 nM T87554 CG9C6J 89765129 IC50 = 0.7 nM T87554 C13GOX 89775209 IC50 = 180 nM T87554 C3N6RU 89775221 IC50 = 70 nM T87554 C69JXR 90034304 IC50 = 131 nM T87554 CDO6N1 90034309 IC50 = 85 nM T87554 C3VJ2W 90034362 IC50 = 620 nM T87554 CB74RS 90034368 IC50 = 71 nM T87554 CE8T5K 90034382 IC50 = 690 nM T87554 CFX7M4 90034390 IC50 = 73 nM T87554 CEG3A4 90035164 IC50 = 9 nM T87554 CG5P9A 90153688 IC50 > 50000 nM T87554 CV64KY 90183363 IC50 > 1000 nM T87554 CL4JO2 90183809 IC50 = 718 nM T87554 CTV52A 90367281 IC50 = 19 nM T87554 CFB75T 90479825 IC50 = 6 nM T87554 CY0UC4 90645194 IC50 > 10000 nM T87554 CV9H8U 90656285 IC50 = 1500 nM T87554 CG7E1U 90656286 IC50 = 1225 nM T87554 CDF9O2 90656287 IC50 = 300 nM T87554 C7EXH8 91755097 IC50 = 11 nM T87554 C37IZB 91755098 IC50 = 140 nM T87554 C7UAK5 91809175 IC50 > 2000 nM T87554 C8RG6H 91827514 IC50 = 40 nM T87554 CVR1I7 91827515 IC50 = 8.2 nM T87554 CAU45T 91971978 IC50 > 30000 nM T87554 C64SIO 92042864 IC50 = 1050 nM T87554 C9BL4M 92045136 IC50 > 22000 nM T87554 CXU1Z2 101043725 IC50 > 2000 nM T87554 CRI0S4 101891768 IC50 > 1000 nM T87554 C9G5TC 102515538 Ki = 9 nM T87554 CM2C3W 105539869 IC50 = 1700 nM T87554 CU4O5Z 112901888 IC50 = 140 nM T87554 C3ECY5 117625437 IC50 = 14 nM T87554 CZC84D 117769161 IC50 = 27 nM T87554 CE7BZ8 117769174 IC50 = 160 nM T87554 CBJ07Q 117769217 IC50 = 70 nM T87554 CXHQ08 117769229 IC50 = 15 nM T87554 CS9WO4 117769234 IC50 = 11 nM T87554 C61VXQ 117769241 IC50 = 15 nM T87554 C1SA9I 117769244 IC50 = 19 nM T87554 C0VY7C 117769271 IC50 = 20 nM T87554 C6O9BT 117769272 IC50 = 47 nM T87554 CSR9B0 117769289 IC50 = 20 nM T87554 C2M9CR 117769307 IC50 = 38 nM T87554 C7FWS3 117769309 IC50 = 7.3 nM T87554 CYWV32 117769339 IC50 = 29 nM T87554 CZV35K 117769346 IC50 = 21 nM T87554 C5V6RG 117769349 IC50 = 80 nM T87554 C4O1PX 117769362 IC50 = 22 nM T87554 CPV4C8 117769365 IC50 = 15 nM T87554 CP3MC5 117769379 IC50 = 17 nM T87554 C8V6LG 117769392 IC50 = 22 nM T87554 C2NBZ8 117769396 IC50 = 17 nM T87554 COV59Y 117769408 IC50 = 49 nM T87554 CXJ3I6 117769409 IC50 = 30 nM T87554 C8LTZ6 117769464 IC50 = 19 nM T87554 C4KL1Y 117769470 IC50 = 14 nM T87554 CQ46WT 117769476 IC50 = 36 nM T87554 CSKO30 117769533 IC50 = 44 nM T87554 C6XC3W 117769575 IC50 = 9 nM T87554 CS95HO 117769592 IC50 = 27 nM T87554 C0PIL5 117769623 IC50 = 25 nM T87554 CO3DA2 117769866 IC50 = 7 nM T87554 CI46CP 117770056 IC50 = 390 nM T87554 C7NI8L 117770083 IC50 = 140 nM T87554 CJ3QC8 117770200 IC50 > 10000 nM T87554 CSD47C 117770482 IC50 = 13 nM T87554 C8SNB9 117770595 IC50 = 910 nM T87554 CJ1V9A 117770654 IC50 = 550 nM T87554 CS8E6M 117770678 IC50 = 1400 nM T87554 CM7X9N 117770754 IC50 = 310 nM T87554 C4CFG6 117770831 IC50 = 830 nM T87554 C0X1EQ 117809257 IC50 = 31 nM T87554 CDUH09 117809287 IC50 = 3.5 nM T87554 C8HYU9 117926195 IC50 > 10000 nM T87554 CGQK96 118115537 IC50 > 10000 nM T87554 C2OX1Q 118115706 IC50 = 2030 nM T87554 CWCO47 118115913 IC50 > 10000 nM T87554 C72LYV 118116131 IC50 > 10000 nM T87554 C4JW5D 118116385 IC50 > 10000 nM T87554 CY0H6Z 118129292 IC50 = 68 nM T87554 CJ1LF6 118129295 IC50 = 331 nM T87554 CA7FL8 118129378 IC50 = 2910 nM T87554 C7ZM6W 118129401 IC50 = 369 nM T87554 CNX7M9 118473558 IC50 > 2000 nM T87554 CK6Z8O 118475621 IC50 = 107 nM T87554 CIVS69 118475644 IC50 = 32 nM T87554 C17FYA 118475649 IC50 = 351 nM T87554 CE49ZI 118475652 IC50 = 51 nM T87554 C65NIK 118475658 IC50 > 3000 nM T87554 C0A9RJ 118475705 IC50 = 17.6 nM T87554 CWQ36P 118475893 IC50 > 3000 nM T87554 CN04RH 118475894 IC50 = 945 nM T87554 C2P0CG 118475938 IC50 = 421 nM T87554 CJYV54 118494221 IC50 = 82.4 nM T87554 CLTV08 118690376 IC50 = 17 nM T87554 CRK6J2 118690573 IC50 = 13 nM T87554 CTR74C 118690690 IC50 = 12 nM T87554 CY7BI2 118706214 IC50 > 10000 nM T87554 C2C0AG 118707521 IC50 > 100000 nM T87554 C2DJA0 118707522 IC50 > 100000 nM T87554 CBF28W 118707523 IC50 > 100000 nM T87554 CQ6ON4 118707525 IC50 > 100000 nM T87554 C38UWP 118707526 IC50 > 100000 nM T87554 C64ZQX 118707543 IC50 > 100000 nM T87554 C7EG0V 118712812 IC50 = 394 nM T87554 C57YED 118712813 IC50 = 59 nM T87554 CX58DI 118716791 IC50 > 30000 nM T87554 CD9X2B 118716796 IC50 > 30000 nM T87554 C2YJ0O 118716797 IC50 > 30000 nM T87554 CL3UO9 118716798 IC50 > 30000 nM T87554 C71BAM 118716799 IC50 > 30000 nM T87554 CU4EL6 118716806 IC50 > 30000 nM T87554 CI5W9H 118720010 IC50 = 44 nM T87554 COQ9S4 118720011 IC50 > 1000 nM T87554 CP0IO9 118722564 IC50 = 4410 nM T87554 C5K2QD 118723914 IC50 = 30 nM T87554 C59YJC 118723915 IC50 = 16 nM T87554 C2ON7Y 118723916 IC50 = 570 nM T87554 C5U8WG 118723917 IC50 = 130 nM T87554 C0ZMR8 118723918 IC50 = 100 nM T87554 C4Z5LJ 118723919 IC50 = 350 nM T87554 C85ELI 118723920 IC50 = 61 nM T87554 CGW49X 118723921 IC50 = 150 nM T87554 CXC8K9 118723922 IC50 = 400 nM T87554 CR5JD8 118723923 IC50 = 110 nM T87554 C9W1BU 118723924 IC50 = 380 nM T87554 CW2G9E 118724201 IC50 > 30000 nM T87554 CXQM59 118727237 IC50 = 8500 nM T87554 C1XE3V 118727239 IC50 = 9500 nM T87554 CU0BP1 118727245 IC50 = 6900 nM T87554 CHT6K9 118728811 Ki > 4000 nM T87554 CUA3Y2 118728812 Ki > 4000 nM T87554 CDQ78G 118728813 Ki = 620 nM T87554 CZ6XL7 118728814 Ki = 270 nM T87554 CMO67K 118728815 Ki = 200 nM T87554 CR2M0Q 118728816 Ki > 4000 nM T87554 C62SCL 118728817 Ki > 4000 nM T87554 CSB30C 118728819 Ki = 840 nM T87554 CV7XU8 118728820 Ki = 390 nM T87554 C3J1EX 118728821 Ki > 4000 nM T87554 CIWB78 118728822 Ki = 1100 nM T87554 CP18SE 118728823 Ki = 240 nM T87554 CM42CA 118728824 Ki > 4000 nM T87554 C9Q7CL 118728825 Ki > 4000 nM T87554 CCR3S0 118728826 Ki = 740 nM T87554 C5NIL4 118729140 IC50 = 1068 nM T87554 C6TP4G 118729141 IC50 = 950 nM T87554 CQJY72 118729142 IC50 = 220 nM T87554 CWNA60 118729861 IC50 = 216 nM T87554 CN2SA5 118734641 IC50 = 293 nM T87554 CF6J5Q 118734642 IC50 = 1044 nM T87554 CMHF86 118734643 IC50 = 686 nM T87554 CUE83V 118734644 IC50 = 246 nM T87554 C67IDL 118734645 IC50 = 558 nM T87554 CFD82L 118734646 IC50 = 1475 nM T87554 C26ZJS 118734647 IC50 = 613 nM T87554 CM5A9U 118734648 IC50 = 547 nM T87554 C7HP6N 118734649 IC50 = 684 nM T87554 CVIN49 118734650 IC50 = 835 nM T87554 CQCX41 118737057 IC50 = 2911 nM T87554 C8JGN7 118868847 IC50 = 888 nM T87554 C3DK1Q 118868914 IC50 = 156 nM T87554 CQ1TL7 118879520 IC50 = 286 nM T87554 CAZO34 118911466 IC50 = 11000 nM T87554 C6VAE4 118911477 IC50 = 51 nM T87554 CRQV39 118911480 IC50 = 130 nM T87554 C5Z0XH 118911481 IC50 = 410 nM T87554 CG0T1W 118911482 IC50 = 2800 nM T87554 COD91F 118911483 IC50 = 15000 nM T87554 C5LYI2 118911484 IC50 = 7800 nM T87554 CA9P3K 118911491 IC50 = 260 nM T87554 CB81YO 118911492 IC50 = 66 nM T87554 C2DG5M 118911497 IC50 = 30000 nM T87554 CI2EU5 118911501 IC50 = 7400 nM T87554 CA3EF6 118911506 IC50 = 160 nM T87554 C9BE2G 118911507 IC50 = 16000 nM T87554 C75DOY 118911508 IC50 = 1400 nM T87554 CZ3D0U 118911512 IC50 = 11000 nM T87554 C1AE4J 118911514 IC50 = 1300 nM T87554 CN53SL 118911517 IC50 = 250 nM T87554 CCX4J8 118911542 IC50 = 1300 nM T87554 C7R0NJ 118911545 IC50 = 4700 nM T87554 CIS3Z5 118911549 IC50 = 5.5 nM T87554 C49PME 118911551 IC50 = 9100 nM T87554 CJT3P9 118911552 IC50 = 98000 nM T87554 CX01BU 118911553 IC50 = 1200 nM T87554 C0TU7V 118911556 IC50 = 470 nM T87554 C0TX7B 118911557 IC50 = 1000 nM T87554 CYI3O6 118911558 IC50 = 150 nM T87554 C28MLV 118911560 IC50 = 930 nM T87554 C49UGI 118911561 IC50 = 1200 nM T87554 C9LD1H 118911562 IC50 = 4500 nM T87554 CTR8D0 118911563 IC50 = 1100 nM T87554 CY5EN8 118911565 IC50 = 30 nM T87554 C84BPW 118911566 IC50 = 36 nM T87554 CT4MJ8 118911570 IC50 = 59 nM T87554 C2AZP5 118911571 IC50 = 1100 nM T87554 C2S7MO 118911575 IC50 = 50 nM T87554 C45HFX 118911579 IC50 = 9100 nM T87554 CCSH64 118911580 IC50 = 6300 nM T87554 CB48OQ 118911581 IC50 = 420 nM T87554 CZY2V6 118911582 IC50 = 13000 nM T87554 C2PA8M 118911583 IC50 = 97 nM T87554 C70XKA 118911584 IC50 = 2500 nM T87554 CD9C1A 118911585 IC50 = 2800 nM T87554 CRZ20W 118911587 IC50 = 180 nM T87554 CTQ4J9 118911588 IC50 = 180 nM T87554 C3QKH8 118911601 IC50 = 150 nM T87554 COY26N 118911635 IC50 = 6500 nM T87554 CL3C9A 118911638 IC50 = 4400 nM T87554 CN4O2C 118911639 IC50 = 480 nM T87554 C9O4WL 118911640 IC50 = 2800 nM T87554 C3SE0K 118911642 IC50 = 1300 nM T87554 C5LHC4 118911643 IC50 = 8.4 nM T87554 CYTV80 121284861 IC50 > 2000 nM T87554 C37DUM 121293882 IC50 > 2000 nM T87554 CXQR89 121294143 IC50 = 1100 nM T87554 C08KEM 122179540 IC50 = 4700 nM T87554 C3AJ4C 122179546 IC50 = 6700 nM T87554 CG0RP7 122179547 IC50 = 2700 nM T87554 C1A0SQ 122179548 IC50 = 5600 nM T87554 C42GSX 122180520 Ki > 4000 nM T87554 CO7D4I 122182021 IC50 = 1300 nM T87554 CY9M5S 122182022 IC50 = 7.3 nM T87554 C2MCH6 122182157 IC50 = 84 nM T87554 CD92SA 122182158 IC50 = 640 nM T87554 CK4A6L 122182159 IC50 = 14 nM T87554 C9OWX5 122186256 IC50 > 10000 nM T87554 C3J6BA 122186261 IC50 > 10000 nM T87554 CZN2V0 122188510 IC50 = 6864 nM T87554 CD62MC 122191616 IC50 = 4.5 nM T87554 CJI3E4 122191617 IC50 = 14 nM T87554 CFU15S 122191618 IC50 = 4.2 nM T87554 CE4F3A 122191619 IC50 = 25 nM T87554 CAC5U1 122191620 IC50 = 210 nM T87554 C8C1PI 122191621 IC50 = 1300 nM T87554 CA0D5W 122191622 IC50 = 570 nM T87554 CZ9K5C 122191623 IC50 = 43 nM T87554 C3NYR0 122191624 IC50 = 450 nM T87554 CRF2K0 122191625 IC50 = 230 nM T87554 CFKD32 122191637 IC50 = 1020 nM T87554 CPY1K9 122191778 IC50 = 2451 nM T87554 C1H4IX 122192065 IC50 = 2200 nM T87554 C98EJO 122192066 IC50 = 20500 nM T87554 CM1XD7 122192067 IC50 = 2900 nM T87554 C0MLH5 122192068 IC50 = 1600 nM T87554 CC4T6A 122192069 IC50 = 3200 nM T87554 CGO6M7 122192070 IC50 = 4100 nM T87554 CBP34K 122192071 IC50 = 2800 nM T87554 CA2TF6 122192072 IC50 = 2700 nM T87554 CFY30Z 122192073 IC50 = 2600 nM T87554 CJ09XF 122192074 IC50 = 2600 nM T87554 C6LS8X 122192075 IC50 = 5900 nM T87554 C7DJA5 122192076 IC50 = 4800 nM T87554 CAS86F 122192079 IC50 = 13500 nM T87554 CG7TP0 122192080 IC50 = 4700 nM T87554 C5K8UM 122192081 IC50 = 1600 nM T87554 CS4XB9 122199230 IC50 = 11900 nM T87554 CNA45R 122362931 IC50 = 113 nM T87554 CV7RT2 123263625 IC50 = 100 nM T87554 CW9BU8 126643886 IC50 = 730 nM T87554 C4BJ8G 126645320 IC50 = 170 nM T87554 CL60VJ 126647240 IC50 = 4400 nM T87554 C1XS8H 126647348 IC50 = 89 nM T87554 CSJ1G7 126647349 IC50 = 19000 nM T87554 C9QCD3 126715362 IC50 = 1770 nM T87554 CNPB25 126715363 IC50 > 30000 nM T87554 CY7US6 126715366 IC50 = 6600 nM T87554 CJS53A 126715367 IC50 = 5010 nM T87554 CX37RN 126715380 IC50 > 15000 nM T87554 C2DQU9 126715387 IC50 > 30000 nM T87554 CH6YP0 126715392 IC50 = 5400 nM T87554 C1QB5R 126715400 IC50 = 1800 nM T87554 CG7YQ2 126715454 IC50 = 322 nM T87554 CO2X6J 126715460 IC50 = 1570 nM T87554 CR9C1G 127030133 IC50 = 150 nM T87554 CU4AJ8 127037981 IC50 = 9620 nM T87554 CA0O1B 127037982 IC50 = 16200 nM T87554 C50NKB 127037983 IC50 > 30000 nM T87554 CF8KQ6 127038326 IC50 = 16200 nM T87554 C5WV8P 127038327 IC50 = 2780 nM T87554 CI8ZB6 127038328 IC50 > 30000 nM T87554 C98DQZ 127038947 IC50 > 17000 nM T87554 CQ4OE5 127039917 IC50 > 22000 nM T87554 CC1XP0 127040339 IC50 = 13900 nM T87554 C8H7JN 127040340 IC50 = 4740 nM T87554 CRQS46 127040341 IC50 > 30000 nM T87554 C3B0AP 127040342 IC50 > 30000 nM T87554 C7KLD9 127040660 IC50 = 10300 nM T87554 C4JF8H 127040661 IC50 = 2270 nM T87554 CC9J7R 127040662 IC50 = 11800 nM T87554 CP1RY4 127040993 IC50 = 2890 nM T87554 C7P5MY 127040994 IC50 = 13100 nM T87554 CB23SC 127041238 IC50 = 14900 nM T87554 CJ7QW5 127041248 IC50 = 9900 nM T87554 C1N6BC 127041249 IC50 = 2700 nM T87554 C5SLH0 127041250 IC50 > 30000 nM T87554 C28YFA 127041251 IC50 > 30000 nM T87554 CIP84Z 127041549 IC50 > 30000 nM T87554 CQP76E 127041550 IC50 > 30000 nM T87554 C3A1VL 127041551 IC50 > 30000 nM T87554 CEJ97D 127041858 IC50 = 1450 nM T87554 C35OPG 127041859 IC50 = 10100 nM T87554 CEN15W 127041860 IC50 = 3040 nM T87554 C4UBE5 127041861 IC50 > 30000 nM T87554 CD1X4L 127045648 IC50 > 1000 nM T87554 CQ76DA 127045649 IC50 > 1000 nM T87554 C4FT6K 127045650 IC50 > 1000 nM T87554 C7Q5YC 127045965 IC50 = 98 nM T87554 C46WVR 127046091 IC50 = 67 nM T87554 C3V5BF 127046092 IC50 = 8 nM T87554 C4SYH9 127046093 IC50 = 21 nM T87554 C5X2VQ 127046094 IC50 = 9 nM T87554 C9YC1K 127046298 IC50 = 78 nM T87554 CQWK04 127046639 IC50 = 732 nM T87554 CZIY10 127046798 IC50 = 531 nM T87554 CX63EC 127046918 IC50 = 184 nM T87554 C6OAX1 127047114 IC50 = 20 nM T87554 CZE85O 127047115 IC50 = 4800 nM T87554 C0R1FI 127047116 IC50 = 1200 nM T87554 CX7LZ6 127047117 IC50 = 908 nM T87554 CAML79 127047118 IC50 > 1000 nM T87554 CCG12W 127047119 IC50 = 155 nM T87554 C2Y1OE 127047142 IC50 = 10 nM T87554 CRYP16 127047143 IC50 = 94 nM T87554 C90NAH 127047271 IC50 = 81 nM T87554 C1UI3Z 127047798 IC50 = 41 nM T87554 CRY8T0 127047799 IC50 = 36 nM T87554 C53OCD 127047800 IC50 = 23 nM T87554 CGA6L4 127047801 IC50 = 6 nM T87554 C26NKY 127047920 IC50 = 17 nM T87554 C19LEF 127047991 IC50 = 97 nM T87554 CS2VY8 127048034 IC50 = 786 nM T87554 CI8Y2P 127048035 IC50 = 475 nM T87554 CB2SE8 127049004 IC50 = 18500 nM T87554 CS6ZO5 127049005 IC50 = 27300 nM T87554 C1PE9L 127050562 IC50 = 3200 nM T87554 CZ5D8C 127050563 IC50 = 29700 nM T87554 CX46RS 127050564 IC50 = 12100 nM T87554 C3LI1J 127050565 IC50 = 3900 nM T87554 CG91WC 127052080 IC50 = 3100 nM T87554 C2LWZ1 129318964 IC50 > 10000 nM T87554 C0FM1R 130196825 IC50 = 170 nM T87554 CZ13WL 130339268 IC50 = 74 nM T87554 CD4NY1 131839645 IC50 = 3.9 nM T87554 C6OXE3 132134663 IC50 = 1.4 nM T87554 CUO0C5 132156633 IC50 > 10000 nM T87554 CV89JM 132231876 IC50 = 3300 nM T87554 CK4FI7 132277003 IC50 > 10000 nM T87554 C5CZA1 132578411 IC50 = 41.9 nM T87554 CDMF97 134130282 IC50 > 100000 nM T87554 C2H6PW 134130554 IC50 = 126 nM T87554 CWF16B 134131331 IC50 = 129 nM T87554 CLV5I3 134131586 IC50 = 50 nM T87554 C5CD9F 134131902 IC50 < 39 nM T87554 CA75NE 134135874 IC50 = 8.9 nM T87554 CR6D9H 134136093 IC50 = 25.7 nM T87554 CQH05W 134136683 IC50 = 18.9 nM T87554 CQ93RF 134136880 IC50 < 39 nM T87554 CG21VI 134136955 IC50 < 39 nM T87554 CDY10C 134137518 IC50 = 136.7 nM T87554 C6VHL4 134137944 IC50 = 324.5 nM T87554 CI0DC7 134138196 IC50 = 6.9 nM T87554 C26PWD 134139689 IC50 = 2.57 nM T87554 C8CP1R 134141659 IC50 = 1.27 nM T87554 CID3G7 134142328 IC50 = 16.6 nM T87554 CFJX74 134142865 IC50 = 1.71 nM T87554 C41ZEF 134143846 IC50 = 7089 nM T87554 C7FXS5 134144592 IC50 = 9 nM T87554 C9Y0KW 134144836 IC50 < 39 nM T87554 CEDU72 134145690 IC50 = 5 nM T87554 C1E2ZW 134145921 IC50 = 4.7 nM T87554 CL9H5I 134146726 IC50 < 39 nM T87554 C8O9SN 134147898 IC50 = 4.3 nM T87554 C48AOM 134150297 IC50 = 10.4 nM T87554 CG9H5W 134150350 IC50 = 2.31 nM T87554 CJX12K 134151832 IC50 = 2.45 nM T87554 CHJ2I6 134152624 IC50 < 39 nM T87554 C96JCY 134153909 IC50 = 30 nM T87554 C4B7IL 134154440 IC50 = 226.1 nM T87554 C8F1BP 134156083 IC50 = 0.97 nM T87554 CCN19D 134157542 IC50 < 39 nM T87554 C1FCZ6 134158025 IC50 = 47 nM T87554 C75NKQ 134537028 IC50 = 1500 nM T87554 CPDT50 134537033 IC50 = 4300 nM T87554 C8CKE5 134537037 IC50 = 1900 nM T87554 C7H8QW 134537039 IC50 = 110 nM T87554 C0ZY5J 134537043 IC50 = 130 nM T87554 CJDM08 134537050 IC50 = 3900 nM T87554 CQ7G4C 134537056 IC50 = 57 nM T87554 CQ1NX6 134537061 IC50 = 27000 nM T87554 C43CFZ 134537067 IC50 = 4800 nM T87554 CELH87 134537071 IC50 = 460 nM T87554 C8DAO7 134537074 IC50 = 18 nM T87554 CQ9OU1 134537081 IC50 = 4500 nM T87554 CH78PN 134537085 IC50 = 1700 nM T87554 CN5P0G 134537092 IC50 = 5900 nM T87554 CHY1S4 134537094 IC50 = 1100 nM T87554 C8L7UN 134537111 IC50 = 110 nM T87554 C42TFN 134537113 IC50 = 690 nM T87554 C58HUF 134537114 IC50 = 1900 nM T87554 C3LRB2 134537119 IC50 = 550 nM T87554 CWU3Z2 134537141 IC50 = 370 nM T87554 CEOW01 134537147 IC50 = 1400 nM T87554 C0T7VN 134537152 IC50 = 2400 nM T87554 CZD72H 134537156 IC50 = 1200 nM T87554 C3HC0S 134537158 IC50 = 240 nM T87554 CTP15L 134537160 IC50 = 3900 nM T87554 C6Z9QY 134537161 IC50 = 430 nM T87554 C9ME6L 134537163 IC50 = 53 nM T87554 CEQ15Z 134537167 IC50 = 4700 nM T87554 C8N6ZF 134537169 IC50 = 3400 nM T87554 CXA39D 134537177 IC50 = 1800 nM T87554 C97OTS 134537185 IC50 = 1300 nM T87554 CHK0V4 134611545 IC50 = 6.6 nM T87554 C20FAE 134611548 IC50 = 83 nM T87554 C51PKU 134611580 IC50 = 5.6 nM T87554 CN75GU 134611727 EC50 = 7710 nM T87554 C80PJI 134611728 IC50 = 48 nM T87554 CFM46L 134812674 IC50 = 366 nM T87554 C2VC5Y 134817793 IC50 = 929 nM T87554 C54FXD 134957362 IC50 > 10000 nM T87554 CVF86X 135125189 IC50 = 3.2 nM T87554 C9MCQ0 135138184 IC50 = 6 nM T87554 C7V2MJ 135142423 IC50 = 2.8 nM T87554 CLET52 135142442 IC50 = 2.1 nM T87554 CU13RW 135142625 IC50 = 7.2 nM T87554 CM7N0J 135142656 IC50 = 22 nM T87554 CG6JI9 135142885 IC50 = 5.6 nM T87554 CQD32R 135143120 IC50 = 9.2 nM T87554 CTJ48K 135524085 IC50 = 3600 nM T87554 CUT1W7 135524168 IC50 = 1300 nM T87554 C7PJ6X 135566704 IC50 > 30000 nM T87554 CI47VJ 135566923 IC50 = 105 nM T87554 CPHG43 135567142 IC50 = 4 nM T87554 C2NRS8 135567293 IC50 = 2.2 nM T87554 C4R1FH 135567294 IC50 = 4.2 nM T87554 CA0R9G 135567295 IC50 = 58.8 nM T87554 CHU3A2 135635724 IC50 = 11000 nM T87554 CPV59N 135685787 Ki > 4000 nM T87554 CRI5F3 135839295 IC50 = 5.4 nM T87554 CH8W7B 135839328 IC50 = 100.8 nM T87554 C29PWN 135886762 IC50 = 3700 nM T87554 CJV08H 135897884 IC50 = 7463 nM T87554 C4K3XL 135897887 IC50 = 551 nM T87554 C93QJC 135897888 IC50 > 10000 nM T87554 CX6JV7 135897894 IC50 = 4410 nM T87554 C5QUL0 135897897 IC50 = 224 nM T87554 CLV7Y8 135897900 IC50 = 589 nM T87554 CFJZ14 135897904 IC50 > 10000 nM T87554 CT2UV5 135897905 IC50 > 10000 nM T87554 CF1PS8 135934877 Ki > 1600 nM T87554 C32BOU 135956049 IC50 = 3 nM T87554 CRU32G 135971388 Ki = 0.8 nM T87554 CTRL59 135976660 Ki = 3500 nM T87554 CJID74 136013449 EC50 = 15800 nM T87554 CHA4N2 136013680 IC50 > 10 nM T87554 C1PCJ3 136042251 IC50 = 830 nM T87554 CHL5Z7 136056540 IC50 = 120 nM T87554 CO0L9T 136056541 IC50 = 190 nM T87554 CLIE18 136056542 IC50 = 1810 nM T87554 CM7V8J 136056543 IC50 > 10000 nM T87554 C64BEV 136056544 IC50 = 83 nM T87554 CP1MX4 136056545 IC50 = 290 nM T87554 C4AR8N 136056546 IC50 = 980 nM T87554 CC10GD 136056547 IC50 = 950 nM T87554 CN1PY3 136056548 IC50 = 184 nM T87554 CI8Y0U 136056549 IC50 > 10000 nM T87554 CY7TJ2 136164051 IC50 = 88 nM T87554 CQ84IZ 136180335 Ki > 4000 nM T87554 CC52HL 136189674 IC50 > 3600 nM T87554 C1YUD0 136219394 IC50 > 10 nM T87554 CIU8W3 136254389 IC50 > 10 nM T87554 C1P6ZW 136263939 IC50 = 0.3 nM T87554 C0R2IL 136901416 IC50 = 6.31 nM T87554 C5JIR2 136987005 IC50 > 100000 nM T87554 CIJ71W 137028350 IC50 = 1300 nM T87554 CS15TL 137028351 IC50 = 2500 nM T87554 CH3M4B 137083628 IC50 > 30000 nM T87554 CJA07O 137083629 IC50 > 30000 nM T87554 C9F8PX 137083630 IC50 > 30000 nM T87554 CE9V4U 137174991 IC50 = 5 nM T87554 CM64UH 137175110 IC50 = 40 nM T87554 C70DIP 137223928 IC50 = 15.9 nM T87554 C9F3KV 137321155 IC50 = 29.6 nM T87554 CJK67W 137321156 IC50 = 3.57 nM T87554 C3Z4AT 137321159 IC50 = 3012 nM T87554 CMY0V2 137321160 IC50 > 6578 nM T87554 CWM9S4 137349398 IC50 = 71 nM T87554 C9I5TJ 137631461 Ki = 900 nM T87554 CAM8K0 137632226 IC50 = 2703 nM T87554 CH9WK1 137632228 IC50 = 11000 nM T87554 C7R2HI 137632648 IC50 = 199 nM T87554 C2I3PY 137633211 IC50 = 658 nM T87554 CJN68H 137633647 IC50 = 538 nM T87554 CF6RH5 137633780 IC50 = 2 nM T87554 C2OC5K 137634207 IC50 = 481 nM T87554 CI1E8V 137634241 IC50 = 236 nM T87554 COE76K 137634328 IC50 = 6.4 nM T87554 C6IU0M 137634461 IC50 = 5 nM T87554 CE4DH3 137635161 IC50 = 770 nM T87554 C6JVG9 137635398 IC50 = 75 nM T87554 CMV38W 137635509 IC50 > 2000 nM T87554 C0VXM3 137635710 Ki = 36 nM T87554 CM73AT 137635759 IC50 = 4670 nM T87554 C63ZFX 137636534 IC50 = 502 nM T87554 CH5SI7 137636771 IC50 = 326 nM T87554 C8FH1S 137637247 IC50 = 200 nM T87554 C8I2NQ 137637573 IC50 = 745 nM T87554 C3RF7B 137638414 IC50 = 1390 nM T87554 CE0ZF8 137638897 IC50 = 5.6 nM T87554 C0J8ZG 137639219 IC50 = 43 nM T87554 C3V4KQ 137641382 IC50 = 219 nM T87554 C50WHR 137641404 IC50 = 377 nM T87554 C2VWE5 137642024 IC50 = 1801 nM T87554 CJ6PU9 137642141 IC50 = 21.2 nM T87554 C0RX1Z 137642404 IC50 = 2.7 nM T87554 CVCM89 137642443 Ki = 3200 nM T87554 CKPB85 137642609 IC50 = 865 nM T87554 C9GDQ6 137642740 IC50 = 2114 nM T87554 CXV15S 137642770 IC50 = 3560 nM T87554 C94ELU 137643208 IC50 > 2000 nM T87554 CO83EQ 137643608 IC50 = 79.6 nM T87554 CQP79B 137643915 IC50 = 788 nM T87554 CGHP09 137645020 IC50 = 0.8 nM T87554 CN34SE 137646319 IC50 > 2000 nM T87554 CI8S5A 137646690 IC50 = 3420 nM T87554 CQYM31 137646825 Ki = 590 nM T87554 CGE91V 137646834 IC50 = 848 nM T87554 CE8SH2 137647292 IC50 = 1270 nM T87554 CUA12V 137647912 Ki = 16 nM T87554 CW6D9H 137648009 IC50 = 1990 nM T87554 C0K5AL 137648444 IC50 = 1200 nM T87554 C9KW2L 137648948 IC50 = 940 nM T87554 CHN7A3 137648975 IC50 = 489 nM T87554 CIB60Q 137649981 IC50 = 7 nM T87554 CF4X3E 137650150 IC50 > 10000 nM T87554 CVHT54 137650515 IC50 = 437 nM T87554 CJQ72A 137650866 IC50 > 10000 nM T87554 CA9K6R 137650880 IC50 = 572 nM T87554 COCF21 137651256 IC50 = 0.5 nM T87554 C3Z7LM 137651481 IC50 = 1.9 nM T87554 CQ27PY 137651710 IC50 = 40.9 nM T87554 CYA52Z 137652173 IC50 = 7 nM T87554 C28QUP 137652864 IC50 > 10000 nM T87554 C6UEB9 137653042 IC50 = 708 nM T87554 CK81UT 137654424 IC50 > 2000 nM T87554 CW6SO7 137654686 IC50 > 3310 nM T87554 CCR5B3 137654793 IC50 = 65 nM T87554 CKM89A 137654900 IC50 = 3.4 nM T87554 C26ONG 137654955 IC50 = 199 nM T87554 CE9OW2 137655154 Ki = 6.6 nM T87554 CVBS03 137656215 IC50 = 0.7 nM T87554 CYWE21 137656346 IC50 = 3.3 nM T87554 C6V3WR 137656619 IC50 = 240 nM T87554 CT1EP3 137656679 IC50 = 17.3 nM T87554 C8VC9A 137657080 IC50 = 7.9 nM T87554 C49GYQ 137658008 IC50 = 244 nM T87554 C59BVH 137658028 IC50 = 2 nM T87554 C6UM5X 137658102 Ki = 370 nM T87554 CO6C8I 137658504 IC50 = 592 nM T87554 CW4CK8 137659037 IC50 = 16 nM T87554 C86KOS 137659382 IC50 = 413 nM T87554 CS61AX 137659496 IC50 > 100000 nM T87554 CR41KW 137660124 IC50 = 0.8 nM T87554 CQ8KF2 137660642 IC50 = 893 nM T87554 CU48TN 137661036 Ki = 150 nM T87554 COMQ54 137661391 IC50 = 939 nM T87554 C5VR2U 137661620 IC50 = 265 nM T87554 CJ52WM 137661888 IC50 = 5437 nM T87554 CO4DP9 137662248 Ki = 14 nM T87554 CU2L5H 138108525 IC50 = 346 nM T87554 C2W0JU 138319690 IC50 > 30000 nM T87554 C28PJZ 138376574 IC50 > 30000 nM T87554 CXV84M 138377596 IC50 = 4 nM T87554 C8X9DR 138584993 IC50 = 109.95 nM T87554 C9NL1M 138585023 IC50 = 0.89 nM T87554 CHX6N7 138585027 IC50 = 3.12 nM T87554 C3RM2Z 138585033 IC50 = 1.07 nM T87554 CBF8S4 138585069 IC50 = 1171 nM T87554 C4O0GC 138585070 IC50 = 17.56 nM T87554 C7KYU3 138585074 IC50 = 140.2 nM T87554 CE5S4Z 138585101 IC50 = 489.65 nM T87554 CM63FA 138585111 IC50 = 14.7 nM T87554 C2U8PZ 138585129 IC50 = 10.55 nM T87554 C0Y2WZ 138585150 IC50 = 72.97 nM T87554 CHMX08 138585151 IC50 = 1.82 nM T87554 CA8N5T 138585156 IC50 = 37.07 nM T87554 CG8TR3 138585164 IC50 = 8.91 nM T87554 C3JR7K 138585184 IC50 > 1000 nM T87554 CQI78V 138585192 IC50 = 37.91 nM T87554 C2UCN9 138605457 IC50 = 14.12 nM T87554 C3RM1U 138605458 IC50 = 229.25 nM T87554 CD4M3W 138605461 IC50 = 63.04 nM T87554 C4VMQ9 138605557 IC50 = 220.8 nM T87554 CQ6R7X 138911330 IC50 = 2700 nM T87554 CI1D9F 139600335 IC50 = 0.7 nM T87554 CI7C4P 140943115 IC50 > 2000 nM T87554 C7U3KH 140943149 IC50 > 2000 nM T87554 C9ZYG8 141366083 IC50 = 5700 nM T87554 C18QDP 141523774 IC50 = 72.3 nM T87554 CD9F4Y 141523776 IC50 = 94.3 nM T87554 C4L6JD 141523781 IC50 = 13.1 nM T87554 CLOI54 141523782 IC50 = 397.4 nM T87554 CDF78Y 141523783 IC50 = 160.3 nM T87554 CSZQ36 141523784 IC50 = 62 nM T87554 CTYQ49 141523785 IC50 = 90.1 nM T87554 C8FC9Y 141531439 IC50 = 469.3 nM T87554 CU51PI 141531440 IC50 = 499 nM T87554 C81RPA 141531442 IC50 = 808.3 nM T87554 CAT46B 141531443 IC50 = 396.2 nM T87554 CS37YV 141531444 IC50 = 1932.5 nM T87554 CEHD51 141728806 IC50 = 12 nM T87554 CCY30N 141728810 IC50 = 22 nM T87554 CLH76T 141728811 IC50 = 20 nM T87554 CQB0U4 141728813 IC50 = 15 nM T87554 CN75MA 141728817 IC50 = 14 nM T87554 CWN43D 141728825 IC50 > 100 nM T87554 C7FW8A 141728827 IC50 = 7 nM T87554 CHS9N0 141728829 IC50 = 21 nM T87554 CN72IC 141728831 IC50 = 10 nM T87554 C7EL5X 141728840 IC50 = 5 nM T87554 C9H8PX 141728841 IC50 = 10 nM T87554 CBV2K5 141728842 IC50 = 36 nM T87554 CZ8J7C 141728843 IC50 = 10 nM T87554 C2HF9A 141728845 IC50 = 61 nM T87554 CBRN42 141728846 IC50 = 46 nM T87554 COEV20 141728855 IC50 > 100 nM T87554 CC03XH 141728860 IC50 = 50 nM T87554 C4RGY1 141728867 IC50 = 46 nM T87554 CNUG79 141728871 IC50 = 30 nM T87554 C65GLX 141728873 IC50 = 5 nM T87554 C9IW0F 141728874 IC50 = 85 nM T87554 C18SJO 141728877 IC50 > 100 nM T87554 CECS13 141753441 IC50 = 1096 nM T87554 C1JR5B 142379949 IC50 = 243 nM T87554 C6C3OH 142744323 IC50 = 156 nM T87554 C45HDA 142744326 IC50 = 96.3 nM T87554 C3SN0Y 142744329 IC50 = 62.7 nM T87554 C2O3RK 142744331 IC50 = 786 nM T87554 C2AWZ6 142744332 IC50 = 210 nM T87554 C4RXO6 142744333 IC50 = 511 nM T87554 CFY17M 142744351 IC50 = 63.6 nM T87554 C5O7KE 142744352 IC50 = 71.8 nM T87554 CM0BL5 142744356 IC50 = 165 nM T87554 C47YDW 142744361 IC50 = 73.5 nM T87554 C2L1ZB 142744367 IC50 = 67.4 nM T87554 CZ6FC4 145362469 IC50 = 450 nM T87554 C6VB3O 145925651 IC50 >= 5000 nM T87554 C2OA9H 145949725 IC50 = 36 nM T87554 CY04PB 145950223 IC50 = 376 nM T87554 CDTW63 145950378 IC50 = 951 nM T87554 CDJ81U 145952312 IC50 = 996 nM T87554 C4BZ0E 145952449 IC50 = 1 nM T87554 C2XP8N 145953005 IC50 > 30000 nM T87554 CA13YG 145953228 IC50 = 16 nM T87554 CN0V3D 145953512 IC50 > 30000 nM T87554 C1OQ3J 145953599 IC50 = 1180 nM T87554 CNS52L 145954024 IC50 = 1030 nM T87554 C4IC5P 145954578 IC50 = 2 nM T87554 CI62ZD 145955000 IC50 = 2 nM T87554 C6QI4B 145955113 IC50 = 8 nM T87554 CRU9F8 145955362 IC50 = 13900 nM T87554 CIP2J9 145955397 IC50 = 357 nM T87554 CZ0K1H 145955759 IC50 = 1 nM T87554 CW2VZ6 145955763 IC50 = 110 nM T87554 CIK4T9 145955799 IC50 = 15 nM T87554 CQ68WS 145956107 IC50 < 3 nM T87554 CZ0B7A 145956262 IC50 = 417 nM T87554 CO6SV3 145957001 IC50 = 6410 nM T87554 C9RH8U 145957804 IC50 = 2 nM T87554 C51ADW 145958260 IC50 = 347 nM T87554 C5XP1C 145958407 IC50 = 3 nM T87554 C3L8IE 145958641 IC50 = 85 nM T87554 C7B2LD 145959014 IC50 = 722 nM T87554 CO05IK 145959360 IC50 = 2 nM T87554 CMCG17 145959462 IC50 = 363 nM T87554 CFC18Z 145960569 IC50 = 18 nM T87554 C2LD5V 145960573 IC50 > 30000 nM T87554 CAGS83 145961653 IC50 = 4 nM T87554 CFY21D 145961655 IC50 = 188 nM T87554 CI9Z7U 145962747 IC50 = 183 nM T87554 CQ86LZ 145963345 IC50 = 765 nM T87554 CPO8J7 145967669 IC50 > 10000 nM T87554 CST35V 145967843 IC50 = 1090 nM T87554 CDNC31 145967951 IC50 > 500 nM T87554 CC3ID7 145968857 IC50 = 3450 nM T87554 C7RF9J 145969339 IC50 = 1420 nM T87554 CWU27Z 145969804 IC50 > 100000 nM T87554 C5VWH3 145970734 IC50 = 46 nM T87554 C63KEL 145970838 IC50 = 3760 nM T87554 CD26ZJ 145970864 IC50 = 1710 nM T87554 C7UG3O 145971121 IC50 = 14100 nM T87554 CEDZ18 145971190 IC50 > 30000 nM T87554 CKPM09 145971514 IC50 = 817 nM T87554 C7K1AJ 145971681 IC50 = 8 nM T87554 CZ85FJ 145972657 IC50 = 1 nM T87554 C7OD0E 145973587 IC50 > 30000 nM T87554 C7TAL5 145979161 IC50 = 41.3 nM T87554 CHVD06 145979212 IC50 > 10000 nM T87554 C7L1IC 145979240 IC50 > 7646 nM T87554 CAJ37B 145979552 IC50 = 1870 nM T87554 CFT50A 145979673 IC50 = 3.4 nM T87554 CE31VG 145979714 IC50 = 1666 nM T87554 C7N8DU 145980127 IC50 = 8623 nM T87554 CWH40Y 145980630 IC50 = 1.8 nM T87554 CX94BD 145980658 IC50 = 9.2 nM T87554 C8AMK1 145980722 IC50 = 1046 nM T87554 C09BPI 145980773 IC50 = 25.6 nM T87554 C81XFH 145980840 IC50 = 4964 nM T87554 C9ZT8Y 145981096 IC50 = 58.3 nM T87554 COG0N1 145981347 IC50 = 239 nM T87554 C85XBC 145981348 IC50 = 470 nM T87554 C2OC6Q 145982084 IC50 = 17 nM T87554 CF8R6Z 145982577 IC50 = 0.96 nM T87554 CHI03D 145982623 IC50 = 0.041 nM T87554 C71AZC 145982856 IC50 = 21 nM T87554 CN4T7U 145982897 IC50 = 2.3 nM T87554 CA7K6C 145983002 IC50 = 40 nM T87554 CEU47V 145983063 IC50 = 867.3 nM T87554 C5VF8P 145983087 IC50 = 508.6 nM T87554 CWS14X 145983289 IC50 = 1397.6 nM T87554 CV28DA 145983327 IC50 = 367.2 nM T87554 CA1LM5 145983443 IC50 = 6.6 nM T87554 CS1GK8 145983460 IC50 = 78.4 nM T87554 CG97VS 145983548 IC50 = 696.8 nM T87554 CML89J 145983552 IC50 = 197.4 nM T87554 CA20KM 145983867 IC50 = 590 nM T87554 CS58RN 145983989 IC50 = 168.4 nM T87554 CJLG54 145984020 IC50 = 0.15 nM T87554 C7THN1 145984160 IC50 = 1118 nM T87554 C30EHD 145984172 IC50 = 2554 nM T87554 CL43AD 145984253 IC50 = 0.04 nM T87554 CODK63 145984420 IC50 = 7.7 nM T87554 CP8J3H 145984569 IC50 = 146.8 nM T87554 C42SJR 145984669 IC50 = 696.8 nM T87554 CLH7K9 145984673 IC50 = 103.5 nM T87554 C67HUC 145984822 IC50 = 590 nM T87554 CXWS04 145984852 IC50 = 3 nM T87554 C2ND4F 145985023 IC50 = 19 nM T87554 CG4U3I 145985120 IC50 = 1420.6 nM T87554 CD1T8G 145985288 IC50 > 1000 nM T87554 C3U9IS 145985565 IC50 = 497.4 nM T87554 C2HXR3 145985769 IC50 = 281.7 nM T87554 CY7X5L 145986106 IC50 = 1947 nM T87554 C03PYD 145986466 IC50 < 1000 nM T87554 C2XPR7 145987380 IC50 = 46 nM T87554 CFH27G 145987566 IC50 = 0.9 nM T87554 CW7V1O 145987719 IC50 > 50000 nM T87554 C8NEY2 145987871 IC50 > 7448 nM T87554 C9ZC0H 145987988 IC50 > 2000 nM T87554 CK6U7Z 145988024 IC50 = 33 nM T87554 C8XBL4 145988088 IC50 = 4.6 nM T87554 C9KJ1A 145988137 IC50 = 97 nM T87554 C0NI8A 145988806 IC50 = 4.3 nM T87554 C9BX4U 145988956 IC50 > 9925 nM T87554 CIVK73 145989244 IC50 > 10000 nM T87554 CI97FM 145989333 IC50 = 2.93 nM T87554 CC8GZ3 145989610 IC50 = 1544 nM T87554 C5I8SR 145989639 IC50 > 10000 nM T87554 CIU9W4 145990027 IC50 > 10000 nM T87554 C3DWZ0 145990496 IC50 > 10000 nM T87554 CTX1A3 145990814 IC50 = 876 nM T87554 CO7F1K 145990990 IC50 = 23 nM T87554 CNG35K 145991262 IC50 > 10000 nM T87554 C0M6LD 145991292 IC50 = 2419 nM T87554 CKGE38 145991618 IC50 = 783 nM T87554 CZ94XS 145991731 IC50 = 18 nM T87554 CJC47L 145992551 IC50 = 95.5 nM T87554 C3RC5J 145992581 IC50 = 2.6 nM T87554 CI8R6P 145992803 IC50 > 10000 nM T87554 CD09RT 145992905 IC50 = 3.1 nM T87554 CG21JZ 145993080 IC50 > 50000 nM T87554 CR2F1Y 145993348 IC50 = 2455 nM T87554 C51DMH 145993445 IC50 > 10000 nM T87554 C51ZNC 145993585 IC50 = 3.9 nM T87554 CF36GI 145993689 IC50 = 109 nM T87554 CSQ7G0 145994254 IC50 = 3.6 nM T87554 C19PRG 145998263 IC50 = 100000 nM T87554 C1S2ER 146025986 IC50 = 2200 nM T87554 CJ8B7I 146185140 IC50 = 48 nM T87554 CHQU21 146185142 IC50 = 26 nM T87554 CS92OU 146185145 IC50 = 119 nM T87554 CXTH86 146185148 IC50 = 35 nM T87554 CP96SV 146185154 IC50 = 461 nM T87554 C71KXB 146185156 IC50 = 16 nM T87554 C9IA1X 146185163 IC50 = 3 nM T87554 CS0OL6 146185170 IC50 = 6 nM T87554 C1IAH7 146185174 IC50 = 27 nM T87554 CXGV39 146185193 IC50 = 37 nM T87554 CZX3B5 146185203 IC50 = 3400 nM T87554 C35CPK 146185546 IC50 = 3049 nM T87554 C5DAO2 149003255 IC50 = 437.1 nM T87554 CZ0LP6 150496562 IC50 = 18 nM T87554 CONR74 154637047 IC50 = 9.3 nM T87554 C7HKA9 154637067 IC50 = 11 nM T87554 CL9P8H 154637078 IC50 = 27 nM T87554 C5T7UA 154701267 IC50 = 24 nM T87554 C7PLT9 155510967 IC50 > 4216 nM T87554 C1WRE2 155511764 IC50 = 2 nM T87554 CR1SE8 155511850 IC50 = 1083 nM T87554 C91YXU 155511860 IC50 = 642.1 nM T87554 CDY5U0 155512704 IC50 = 182 nM T87554 CT9B4M 155512787 IC50 = 437 nM T87554 C2MD1Q 155513187 IC50 > 10000 nM T87554 CM95KR 155513637 IC50 = 396.4 nM T87554 C83ZSG 155514311 IC50 = 160 nM T87554 C7MJY5 155514805 IC50 = 45 nM T87554 CUIO35 155516044 IC50 = 11.5 nM T87554 CD6YR0 155516192 IC50 = 870.4 nM T87554 CTP29J 155516678 IC50 = 2.4 nM T87554 C9VK3I 155517004 IC50 > 50000 nM T87554 C2X8HA 155517088 IC50 > 50000 nM T87554 CE2Q3D 155517448 IC50 = 380 nM T87554 C0E7WS 155518120 IC50 = 692 nM T87554 CDTG10 155518349 IC50 = 5 nM T87554 CQ19HO 155518921 IC50 = 560 nM T87554 CLK4S9 155519594 IC50 = 411 nM T87554 CF0H9V 155520176 IC50 = 503 nM T87554 C0A9LX 155520276 IC50 > 10000 nM T87554 C4YJN9 155520341 IC50 = 77 nM T87554 C1PJC7 155520619 IC50 > 30000 nM T87554 C0YEX7 155521332 IC50 = 370 nM T87554 CLZ08K 155522634 IC50 = 604.7 nM T87554 CXG4L3 155522806 IC50 = 2 nM T87554 CEU10G 155522970 IC50 = 112 nM T87554 C9LUO3 155523352 IC50 = 2500 nM T87554 C7NVQ5 155523535 IC50 = 6.5 nM T87554 C32POG 155523862 IC50 = 57.2 nM T87554 C1HWG6 155524274 IC50 = 102 nM T87554 CU7EQ5 155525897 IC50 = 29.8 nM T87554 CE4FX7 155525956 IC50 = 14.8 nM T87554 C39EGQ 155526165 IC50 = 589.5 nM T87554 CCS24O 155527492 IC50 = 82.1 nM T87554 CK14UT 155528172 IC50 = 2782 nM T87554 CB26JT 155528364 IC50 = 110 nM T87554 CVW07K 155528897 IC50 = 3 nM T87554 CMIC15 155529301 IC50 = 35.4 nM T87554 CL47NH 155529550 IC50 = 1800 nM T87554 CX0B9Q 155530477 IC50 = 5.8 nM T87554 CT9R6V 155530931 IC50 = 65 nM T87554 C67TQL 155530972 IC50 = 194 nM T87554 CRX08F 155531665 IC50 > 30000 nM T87554 CQU09F 155532106 IC50 = 30000 nM T87554 C5V6PY 155532206 IC50 > 2000 nM T87554 C4LE7Q 155532724 IC50 = 30 nM T87554 C75AKY 155533695 IC50 > 2000 nM T87554 CLSV71 155533995 IC50 = 1700 nM T87554 CGH63O 155534464 IC50 = 4 nM T87554 CM0U3I 155534552 IC50 > 1000 nM T87554 C2NPE6 155534808 IC50 = 220 nM T87554 C64FIW 155534972 IC50 = 3148 nM T87554 CE8QW2 155535975 IC50 = 50 nM T87554 C2CG1A 155537016 IC50 > 10000 nM T87554 C06JDH 155537151 IC50 = 190 nM T87554 CMV7B2 155538485 IC50 > 30000 nM T87554 C5GNH8 155538704 IC50 = 2790 nM T87554 C5WB0T 155539358 IC50 = 3540 nM T87554 C03BNT 155539537 IC50 = 3230 nM T87554 C3O6KI 155540160 IC50 = 345 nM T87554 C0D8OL 155540191 IC50 = 7.943 nM T87554 C16MHE 155540242 IC50 > 2000 nM T87554 CBA08W 155540345 IC50 = 820 nM T87554 CP2NY0 155540484 IC50 = 5.012 nM T87554 CF8O5T 155540488 IC50 = 3162.28 nM T87554 C51JNT 155540621 IC50 = 10 nM T87554 C5BTX7 155540994 IC50 = 985.9 nM T87554 C76QBR 155541045 IC50 > 30000 nM T87554 CT1AX5 155541077 IC50 = 7.943 nM T87554 CY8F7S 155541097 IC50 = 538 nM T87554 CH6LV1 155541475 IC50 = 19.95 nM T87554 CS58BA 155541478 IC50 = 1444 nM T87554 CF9AX3 155542099 IC50 = 24 nM T87554 C1B6EK 155542401 IC50 = 25.12 nM T87554 CH59RW 155542578 IC50 = 67 nM T87554 CKL31P 155542961 IC50 = 158.49 nM T87554 CH46TG 155543289 IC50 > 3000 nM T87554 C1QRZ2 155543349 IC50 = 146 nM T87554 CRA21U 155543538 IC50 = 916 nM T87554 CD9Z3W 155544141 IC50 = 2.3 nM T87554 CWSG67 155544202 IC50 = 914.5 nM T87554 CZ3YI6 155544372 IC50 = 583 nM T87554 CTQ63L 155544706 IC50 = 19.95 nM T87554 CP7XE1 155545114 IC50 = 19.95 nM T87554 CFR42U 155545338 IC50 = 158.49 nM T87554 C5BHW8 155546008 IC50 = 18 nM T87554 C5U8HP 155546232 IC50 = 10 nM T87554 CJ8F7V 155546474 IC50 = 6340 nM T87554 CO7ZM2 155546902 IC50 = 13.8 nM T87554 CSI1U9 155547916 IC50 = 260 nM T87554 C0B3RK 155547921 IC50 = 199.53 nM T87554 C3DZU0 155548345 IC50 = 200 nM T87554 C67AYP 155548399 IC50 = 28.8 nM T87554 CPR01A 155549631 IC50 = 126 nM T87554 CI6Y5Z 155549690 IC50 = 7.943 nM T87554 CO6ID4 155550122 IC50 = 43 nM T87554 C10OSG 155550219 IC50 = 190 nM T87554 C3DW8J 155550308 IC50 = 15.85 nM T87554 C31QUW 155550462 IC50 = 25 nM T87554 C6UJS7 155550600 IC50 = 240 nM T87554 C2RQT8 155550913 IC50 > 500 nM T87554 C0DMP2 155551420 IC50 = 2098 nM T87554 CHM8G1 155551600 IC50 = 1970 nM T87554 CX0HL6 155552133 IC50 = 1162.8 nM T87554 C2Q1LR 155552255 IC50 = 2400 nM T87554 CW1UX0 155552333 IC50 = 19.95 nM T87554 CV4NX3 155552736 IC50 = 1540 nM T87554 C62ERW 155552853 IC50 = 79.43 nM T87554 CPB6M8 155553409 IC50 = 1015 nM T87554 C5HQ7X 155553551 IC50 = 57 nM T87554 CADO35 155554376 IC50 = 38 nM T87554 CNTP52 155554413 IC50 = 306 nM T87554 CWLC85 155554605 IC50 = 7.2 nM T87554 CQ6S8E 155554939 IC50 = 19.95 nM T87554 C47MNG 155554972 IC50 > 30000 nM T87554 CP39ZD 155555305 IC50 = 125.89 nM T87554 C28MLB 155555377 IC50 = 15200 nM T87554 C9J4HM 155555486 IC50 = 7851 nM T87554 CTRV23 155555922 IC50 > 30000 nM T87554 CG48UE 155556474 IC50 = 10 nM T87554 C8TYG7 155556520 IC50 > 10000 nM T87554 C59HKP 155557055 IC50 > 3000 nM T87554 CZUT98 155557375 IC50 = 28 nM T87554 CG9E7Z 155557901 IC50 = 23 nM T87554 CHW4O3 155558352 IC50 = 7.943 nM T87554 C7HFI8 155558403 IC50 = 1 nM T87554 C7WND0 155558729 IC50 = 684 nM T87554 C3V5HL 155559143 IC50 = 9.7 nM T87554 C2U5ZM 155559343 IC50 = 25.12 nM T87554 CANJ25 155559746 IC50 = 1000 nM T87554 C46KLS 155559780 IC50 = 45.3 nM T87554 CNK81M 155560413 IC50 = 31.62 nM T87554 C54NQC 155561203 IC50 = 488 nM T87554 C1Z6IL 155561218 IC50 = 350 nM T87554 CRU0K3 155563465 IC50 = 3250 nM T87554 C68TCL 155563799 IC50 = 2043 nM T87554 C8HN2B 155563943 IC50 = 36 nM T87554 C1NM2T 155564180 IC50 = 101 nM T87554 CBQN81 155564466 IC50 > 3000 nM T87554 CZ2NK9 155565077 IC50 = 1995.26 nM T87554 CA0Z1U 155565486 IC50 = 1680 nM T87554 CSNF76 155565806 IC50 = 19.95 nM T87554 CF1X5I 155566525 IC50 = 329 nM T87554 C7S5MC 155566661 IC50 > 3000 nM T87554 CQA46B 155566981 IC50 = 2780 nM T87554 CQ5ZX3 155567095 IC50 = 76600 nM T87554 CSRZ04 155567801 IC50 = 280 nM T87554 CGX28M 155567987 IC50 > 30000 nM T87554 COS7X5 155568028 IC50 = 73.1 nM T87554 COGC41 155568181 IC50 = 8 nM T87554 C0L6UT 155568261 IC50 = 19.95 nM T87554 CR79DJ 155568314 IC50 = 366 nM T87554 CRHE56 155569596 IC50 = 9530 nM T87554 CE50IC 155569626 IC50 = 2000 nM T87554 C3X6WU 155569641 IC50 = 718 nM T87554 C14DIR 16750188 IC50 = 130 nM T87554 C5UI4F 16750189 IC50 = 260 nM T87554 C6JKT9 16750206 IC50 = 230 nM T87554 CYIU14 16750228 IC50 = 24 nM T87554 CX4I6T 16750253 IC50 = 36 nM T87554 CI79TY 16750254 IC50 = 60 nM T87554 CS6UT4 16750288 IC50 = 41 nM T87554 COM3C1 16750290 IC50 = 25 nM T87554 CI67WG 16750292 IC50 = 7 nM T87554 CIGJ63 16750308 IC50 = 77 nM T87554 CL2SY5 16750330 IC50 = 330 nM T87554 CE5P2I 53363072 IC50 = 83 nM T87554 CTV60O 53363073 IC50 = 84 nM T87554 CD74BW 53363074 IC50 = 120 nM T87554 CU3M8P 53363075 IC50 = 150 nM T87554 C07FTA 53363076 IC50 = 220 nM T87554 C9JX2G 53363150 IC50 = 15 nM T87554 CJ04SF 53363151 IC50 = 22 nM T87554 CO7Z2P 53363152 IC50 = 22 nM T87554 C1T2LY 53363154 IC50 = 48 nM T87554 C9GEA7 53363242 IC50 = 96 nM T87554 CA06ID 53363244 IC50 = 35 nM T87554 CTSP38 53363245 IC50 = 44 nM T87554 CM7BZ3 53363246 IC50 = 17 nM T87554 C0QON7 53363337 IC50 = 24 nM T87554 CU76JB 53363338 IC50 = 19 nM T87554 C2PU3M 53364335 IC50 = 1200 nM T87554 C10FXI 53364337 IC50 = 70 nM T87554 C2U9QE 53364338 IC50 = 53 nM T87554 D00ERW 44444843 Ki > 1453 nM T87554 D00HVA 11624601 Ki > 1500 nM T87554 D02BXJ 46864270 IC50 = 536 nM T87554 D02NNT 53232451 IC50 < 1 nM T87554 D03BQI 3794 IC50 > 10000 nM T87554 D04NGS 5330790 IC50 = 2960 nM T87554 D05MHL 44605611 Ki = 0.001 nM T87554 D06HVH 54613583 IC50 > 10000 nM T87554 D07OXC 11650194 IC50 > 25000 nM T87554 D08HFG 24809764 IC50 = 3200 nM T87554 D09HVH 135566652 IC50 > 10 nM T87554 D0D6MH 11617559 IC50 > 13000 nM T87554 D0E0XV 9903786 Ki = 5 nM T87554 D0E5IP 3795 IC50 > 10000 nM T87554 D0E7VO 59627005 IC50 = 68.3 nM T87554 D0GN5Z 5281295 IC50 = 9320 nM T87554 D0H7DQ 6419755 IC50 = 3850 nM T87554 D0I3EY 11492186 IC50 = 1600 nM T87554 D0IR6U 5494425 IC50 = 1 nM T87554 D0J3LR 11634725 Ki > 4000 nM T87554 D0K5UF 72710568 IC50 = 12 nM T87554 D0ME9B 46868971 IC50 > 10 nM T87554 D0OP3D 25099184 Ki = 0.45 nM T87554 D0P6JS 11675054 IC50 > 10000 nM T87554 D0Q3NG 11715520 Ki > 1500 nM T87554 D0R2WK 16038120 IC50 = 1505 nM T87554 D0S7IE 11658882 Ki > 1500 nM T87554 D0US9O 45275255 IC50 < 3 nM T87554 D0V6VQ 53344620 IC50 = 123.6 nM T87554 D0VC0I 5169 IC50 > 100000 nM T02001 D07ESC 11561674 IC50 = 33 nM T02001 D0NJ3V 4680 IC50 = 1400 nM T02001 D0R4UW 449193 IC50 = 0.2 nM T02001 D0Z7ZM 135398744 IC50 = 20000 nM T02001 D01LCC 17754438 IC50 > 10000 nM T02001 D03QJL 3671 IC50 = 166 nM T02001 D04XVJ 66829720 IC50 = 5 nM T02001 D09TFB 9896267 IC50 = 13 nM T02001 D0IZ8X 90111638 IC50 = 127 nM T02001 D0LI1C 44469321 IC50 > 10000 nM T02001 D0M7CB 9919680 IC50 = 5.1 nM T02001 D0SM0W 44591583 IC50 = 55 nM T02001 D0T5PO 5092 IC50 = 31.6 nM T02001 D0Z2FB 154575 IC50 = 0.021 nM T02001 D05VBJ 71295299 IC50 = 5890 nM T02001 D0WS3T 72706254 IC50 = 9300 nM T02001 D00YPW 135399235 Ki = 8760 nM T02001 D02EMR 151170 IC50 = 11 nM T02001 D06ABW 2788 IC50 > 10000 nM T02001 D08SNX 135430158 Ki = 141 nM T02001 D0BK6B 3021729 Ki > 50000 nM T02001 D0F0CS 5723 IC50 = 160 nM T02001 D0UG4T 127928 IC50 = 2.1 nM T02001 C1O0CE 40409 IC50 = 1500 nM T02001 C4B3YS 78864 IC50 = 622 nM T02001 C1H8NR 155248 IC50 = 26000 nM T02001 CYS06W 156149 IC50 = 3590 nM T02001 CSO8Q2 176911 IC50 = 6820 nM T02001 CYWS98 185848 IC50 = 2910 nM T02001 C1AN5Z 215436 IC50 = 82000 nM T02001 CZT08K 290897 IC50 = 1870 nM T02001 C1SRY2 529893 IC50 > 20000 nM T02001 CH3FB8 618370 IC50 = 960 nM T02001 CT95PB 656964 IC50 = 270 nM T02001 CY39ZN 656965 IC50 = 2000 nM T02001 CZE5R6 656966 IC50 = 160 nM T02001 C29DYI 656969 IC50 = 21 nM T02001 C1B6ZL 662965 IC50 = 18 nM T02001 CM0Q1K 675863 IC50 = 6309.57 nM T02001 CX40IM 791888 IC50 = 645.65 nM T02001 CM86KB 826384 IC50 = 1900 nM T02001 CR35EF 832190 IC50 = 2300 nM T02001 C75VMR 1047282 IC50 = 100 nM T02001 C7N3SZ 1130142 IC50 = 965 nM T02001 C09ZDF 1158635 IC50 = 380 nM T02001 C8G2PE 1506612 IC50 = 21300 nM T02001 C8JLO0 2243267 IC50 = 3900 nM T02001 CLX0W5 2566813 IC50 = 77200 nM T02001 CW57NL 2852188 IC50 = 501.19 nM T02001 CY7IG8 2853935 IC50 > 2511.89 nM T02001 CVJ36Q 2862736 IC50 > 2511.89 nM T02001 C4LSR7 2886111 IC50 = 316.23 nM T02001 CHV64Q 3713518 IC50 = 604 nM T02001 CK12OT 3814427 IC50 > 20000 nM T02001 CV0AQ4 4198517 IC50 = 2780 nM T02001 C7HST8 4231279 IC50 = 6309.57 nM T02001 CL1Q4X 4254532 IC50 = 52 nM T02001 CB73HU 4398380 IC50 = 125.89 nM T02001 CC3LA4 4672917 IC50 = 470 nM T02001 C5P0LU 4672918 IC50 = 1700 nM T02001 C12SRB 5214710 IC50 = 125.89 nM T02001 C0D3PO 5281671 IC50 = 900 nM T02001 C2MW1L 5319924 IC50 = 260 nM T02001 C8CKQ1 5321960 IC50 = 9980 nM T02001 CH6DT9 5481958 IC50 = 310 nM T02001 C8OAX1 6440408 IC50 = 1260 nM T02001 CJPQ16 6603746 IC50 = 631 nM T02001 CJ8EA9 6918641 IC50 = 11880 nM T02001 C6G4QC 6918642 IC50 = 33330 nM T02001 CI7K0P 6918667 IC50 = 1420 nM T02001 CP1GO7 6918668 IC50 = 1460 nM T02001 CH7QO4 6918791 IC50 > 101000 nM T02001 CEBY83 6918792 IC50 = 92330 nM T02001 C87WYR 6918795 IC50 = 1630 nM T02001 CRGE51 6918796 IC50 = 1590 nM T02001 CUP4M8 6918797 IC50 = 1500 nM T02001 C0LRO8 6918798 IC50 = 15000 nM T02001 C53ESK 6918799 IC50 = 12200 nM T02001 CU1E0G 6918800 IC50 = 7350 nM T02001 CNC2F4 9798336 IC50 = 70.79 nM T02001 CFJ62Y 9799389 IC50 = 1.5 nM T02001 CYXD04 9810934 IC50 = 9 nM T02001 CB7QD5 9827600 Ki = 0.06166 nM T02001 CP9C4H 9835391 IC50 = 6300 nM T02001 C2VLX0 9835752 IC50 = 81500 nM T02001 C4J2XE 9836643 IC50 = 13000 nM T02001 C6HV9M 9836880 IC50 > 101000 nM T02001 CL70YN 9840066 IC50 = 2.7 nM T02001 C18EZT 9857161 IC50 = 22170 nM T02001 CN1YU0 9857760 IC50 = 57000 nM T02001 CA23EP 9858103 IC50 = 15300 nM T02001 CAY84B 9869820 IC50 = 0.85 nM T02001 C0Q5VN 9880010 IC50 > 101000 nM T02001 CWD1F6 9880288 IC50 = 53200 nM T02001 CC05QE 9901606 IC50 > 101000 nM T02001 CJG9R8 9904574 IC50 = 660 nM T02001 CBA29H 9922545 IC50 = 1700 nM T02001 CKF4C2 9922691 IC50 = 10500 nM T02001 C70AMC 9924305 IC50 = 21330 nM T02001 CKI6N2 9924468 IC50 = 320 nM T02001 C76RTB 9924539 IC50 = 32 nM T02001 C6AZ5F 9924709 IC50 = 12000 nM T02001 C81LSK 9928390 IC50 = 4 nM T02001 CA1S6U 9946483 IC50 = 25000 nM T02001 CX1UV7 9946954 IC50 = 23000 nM T02001 C7OP5A 9947052 IC50 = 7050 nM T02001 CM76QK 9966726 IC50 = 22250 nM T02001 CJO0X4 9966737 IC50 > 101000 nM T02001 CFP1Y5 9966830 IC50 > 101000 nM T02001 C0XJ1N 9966833 IC50 > 101000 nM T02001 C9NKY4 9967652 IC50 = 3280 nM T02001 CI6AX1 9968005 IC50 = 44500 nM T02001 C7PCS8 9968050 IC50 > 101000 nM T02001 CFB48Q 9968370 IC50 = 23700 nM T02001 CU73AJ 9968471 IC50 = 99000 nM T02001 C0AP8O 9969020 IC50 = 39660 nM T02001 CW6TD3 9973904 IC50 = 22 nM T02001 CV6TO1 9995407 IC50 = 15.6 nM T02001 CA9YF5 9998837 IC50 = 19 nM T02001 CFPR64 9999276 IC50 = 1 nM T02001 C53HZC 9999401 IC50 = 51 nM T02001 C3A6RV 10027487 IC50 = 0.57 nM T02001 CC86GR 10042087 IC50 = 17 nM T02001 CSK1B0 10046907 IC50 = 5510 nM T02001 CA9Y7L 10066910 IC50 = 8 nM T02001 CJ16FV 10087963 IC50 = 10715.19 nM T02001 C2YV5D 10089968 IC50 = 398.11 nM T02001 C8T3LV 10090103 IC50 = 45 nM T02001 C6T4JS 10091127 IC50 = 51 nM T02001 CT98XQ 10105863 IC50 = 2380 nM T02001 CSI29C 10109508 IC50 = 30 nM T02001 C12LED 10109572 IC50 = 55000 nM T02001 CK5C9Z 10119563 IC50 = 0.7 nM T02001 C1EVS3 10119564 IC50 = 0.5 nM T02001 C83BSD 10128917 IC50 = 0.3 nM T02001 CWDR26 10129145 IC50 = 1.4 nM T02001 C2PBD6 10131447 IC50 = 1550 nM T02001 C8NT0W 10131621 IC50 = 19000 nM T02001 CJ24HR 10132715 IC50 = 15050 nM T02001 CME68G 10152836 IC50 = 0.1 nM T02001 C0PVT2 10153372 IC50 = 1.7 nM T02001 C7D5IT 10158829 IC50 = 24 nM T02001 CBT4P1 10177031 IC50 = 13 nM T02001 C5HC2X 10182563 IC50 = 1310 nM T02001 C3X9DK 10183196 IC50 = 38 nM T02001 CUXV40 10183769 IC50 = 0.5 nM T02001 CY9HS7 10185841 IC50 = 0.2 nM T02001 CVUZ36 10195164 IC50 = 2 nM T02001 C8LYH6 10196396 IC50 = 0.3 nM T02001 CSQ16M 10196596 IC50 = 0.5 nM T02001 CTV6F9 10196609 IC50 = 0.1 nM T02001 CTZ7Q8 10196916 IC50 = 0.8 nM T02001 CZG54F 10197046 IC50 = 0.7 nM T02001 CE5LH4 10199681 IC50 = 6 nM T02001 C3GN8K 10200432 IC50 = 1130 nM T02001 C61CZK 10205978 IC50 = 45 nM T02001 CPU09I 10210579 IC50 = 2.3 nM T02001 CFGO46 10221904 IC50 = 2410 nM T02001 CX9LV3 10232106 IC50 = 1.9 nM T02001 C5T4BP 10246912 IC50 = 13 nM T02001 C7MQZ1 10249183 IC50 = 28.18 nM T02001 CI5Y3F 10254618 IC50 = 0.88 nM T02001 CQ61CV 10268304 IC50 = 1800 nM T02001 C1QU2B 10268305 IC50 = 1010 nM T02001 CH9C4K 10269859 IC50 = 20500 nM T02001 C7RH4B 10270013 IC50 = 64 nM T02001 CR92JY 10270352 IC50 = 14700 nM T02001 C7CHR0 10270536 IC50 = 740 nM T02001 C48ENU 10289786 IC50 = 6.7 nM T02001 CT5FL2 10289848 IC50 = 0.1 nM T02001 CECW14 10301548 IC50 = 0.2 nM T02001 C5IF9A 10312566 IC50 = 0.5 nM T02001 CC7WQ2 10315987 IC50 = 400 nM T02001 CB71WD 10322207 IC50 = 22 nM T02001 C7Z3XL 10335911 IC50 = 3 nM T02001 C52EPV 10339653 IC50 = 3090.3 nM T02001 CJ7YZ9 10345293 IC50 = 0.32 nM T02001 C94EQM 10403778 IC50 = 1584.89 nM T02001 C9A1JH 10432102 IC50 = 30 nM T02001 C23HSK 10451184 IC50 = 2 nM T02001 CD09NL 10451631 IC50 = 30 nM T02001 C1RG7I 10545177 IC50 = 70 nM T02001 C7G1BH 10547592 IC50 = 2000 nM T02001 CZ15HV 10571743 IC50 = 72 nM T02001 C8RN0L 10611778 IC50 = 1600 nM T02001 CHU62M 10661230 IC50 = 7 nM T02001 CRJ79L 10664015 IC50 = 3 nM T02001 CO4AP8 10682163 IC50 = 4100 nM T02001 CIA5D7 10685727 IC50 = 38000 nM T02001 CF2BR1 10691724 IC50 = 48 nM T02001 CNB35R 10805427 IC50 = 8 nM T02001 CDL73U 10810934 IC50 = 11 nM T02001 C0A7DI 11017241 IC50 = 43 nM T02001 CEK01S 11044358 IC50 = 85 nM T02001 C60MEI 11138678 IC50 = 58500 nM T02001 CDJ60K 11229837 IC50 > 20000 nM T02001 C45VZC 11438405 IC50 > 16000 nM T02001 CQ8G9F 11525525 IC50 = 7.9 nM T02001 CS5U1Z 11532316 IC50 = 25 nM T02001 C6UMB2 11532832 IC50 = 11 nM T02001 CX0FM3 11547713 IC50 = 0.7 nM T02001 CE24AU 11626787 IC50 = 128 nM T02001 C0BD7Q 11628421 IC50 = 19 nM T02001 C37TWP 11633996 IC50 = 32 nM T02001 COLF16 11639342 IC50 = 800 nM T02001 C8U5VK 11641556 IC50 = 4.6 nM T02001 C8EX6Z 11648288 IC50 = 13 nM T02001 C83NLR 11648915 IC50 = 61 nM T02001 CX2ZD7 11650267 Ki = 2 nM T02001 CFM64H 11662453 IC50 = 39 nM T02001 CV7E9J 11679574 IC50 = 6568 nM T02001 CQPW60 11705339 IC50 = 3.1 nM T02001 C0I5BW 11711290 IC50 = 34 nM T02001 CVJ10R 11713455 IC50 = 39 nM T02001 C8B4MQ 11742872 IC50 = 40 nM T02001 CROY49 11754228 IC50 = 0.54 nM T02001 CC92YE 11755033 IC50 = 0.53 nM T02001 C1B4XD 11992634 IC50 = 1210 nM T02001 CH9P7X 12000774 IC50 = 0.9 nM T02001 C6MG9U 12000776 IC50 = 8.2 nM T02001 CJ92PF 12000777 IC50 = 1.3 nM T02001 C3BQE0 12000858 IC50 = 0.9 nM T02001 CI5N8Z 12000861 IC50 = 0.7 nM T02001 C7O0WX 12000862 IC50 = 1.4 nM T02001 C51MHW 12000950 IC50 = 1.3 nM T02001 CZF9E8 12112042 IC50 = 2200 nM T02001 C4SRJ0 14521039 IC50 > 20000 nM T02001 C5K2ZP 14521043 IC50 > 20000 nM T02001 C5SM8C 15233693 IC50 = 2330 nM T02001 C40KZA 15434926 IC50 = 70 nM T02001 CVR73F 15549302 IC50 = 26000 nM T02001 C4ESY5 15942639 IC50 = 0.4 nM T02001 C07XUL 15950810 IC50 = 990 nM T02001 CN3I4Z 15950948 IC50 = 1600 nM T02001 C3BI9R 15951010 IC50 = 1700 nM T02001 CWH1A8 15951076 IC50 = 3100 nM T02001 C6VN5F 16067799 IC50 = 13 nM T02001 CMB3Z5 16067906 IC50 = 0.1 nM T02001 C31LJY 16103072 IC50 = 180 nM T02001 C8W2YO 16664188 IC50 = 1000 nM T02001 CXFT59 17757146 IC50 = 49.2 nM T02001 CBX29P 17989733 IC50 = 41 nM T02001 CG4D0L 18436679 IC50 = 0.78 nM T02001 C1PZ8C 18734933 IC50 = 1 nM T02001 C9DE6Y 20814950 IC50 = 4.4 nM T02001 CKAX08 20873492 IC50 = 4320 nM T02001 C3M5NF 21865580 IC50 = 3 nM T02001 C4CWR6 21865595 IC50 = 10 nM T02001 C6T5NZ 21865599 IC50 = 1.9 nM T02001 CULE52 21865620 IC50 = 0.7 nM T02001 CINH54 21865627 IC50 = 2.8 nM T02001 CY06TV 21920178 IC50 = 25750 nM T02001 CL30BY 21920189 IC50 = 5840 nM T02001 C15BGX 21920191 IC50 = 10970 nM T02001 CMZ5G9 21920202 IC50 = 19250 nM T02001 CIB31Y 21920218 IC50 = 34250 nM T02001 CL4R5H 21920232 IC50 = 32250 nM T02001 C68RSV 21920245 IC50 = 8770 nM T02001 C76SHB 21920252 IC50 = 26000 nM T02001 CA2LZ9 21920253 IC50 > 101000 nM T02001 C7RK1W 21920272 IC50 = 14200 nM T02001 CH7N9S 21920275 IC50 = 4260 nM T02001 CBPD46 21920277 IC50 = 19330 nM T02001 C90EXZ 21920288 IC50 = 5900 nM T02001 CWHX89 21920307 IC50 = 44660 nM T02001 CIRD07 21920317 IC50 = 37000 nM T02001 CW5MP2 21920319 IC50 = 17000 nM T02001 CEDO71 21920329 IC50 > 101000 nM T02001 C18YNU 21920341 IC50 > 101000 nM T02001 C0JOK1 21920350 IC50 = 40000 nM T02001 CRN3H8 21920369 IC50 > 101000 nM T02001 CV04DH 21920370 IC50 = 36330 nM T02001 C78SFX 21920385 IC50 > 101000 nM T02001 CMHF08 22083604 IC50 = 2 nM T02001 C34FLM 22083724 IC50 = 0.19 nM T02001 CWIT18 22083784 IC50 = 0.6 nM T02001 C2X0TW 22337167 IC50 = 2.3 nM T02001 CR4T9J 22337182 Ki = 6.3 nM T02001 CFAQ86 22343616 IC50 = 7300 nM T02001 CX0D4Q 22734050 IC50 = 110 nM T02001 CV5C8E 23204708 IC50 = 37153.52 nM T02001 CD48PX 23218492 IC50 = 20.2 nM T02001 CXB78L 23624298 IC50 = 42 nM T02001 C4S6VD 23654252 IC50 = 3467.37 nM T02001 C5J4IN 24774752 IC50 = 190 nM T02001 COC4L2 24774753 IC50 = 30 nM T02001 C7CGN6 24774754 IC50 = 13 nM T02001 CNJ6B0 24774756 IC50 = 100 nM T02001 CG1MF9 24774839 IC50 = 48 nM T02001 CZM0J4 24774840 IC50 = 46 nM T02001 C1FCU4 24774841 IC50 = 25 nM T02001 C51ZNR 24774842 IC50 = 6 nM T02001 C4X5EC 24774843 IC50 = 200 nM T02001 CW9PY5 24774844 IC50 = 29 nM T02001 C1OEA7 24774929 IC50 = 9 nM T02001 CQ6SA9 24774930 IC50 = 40 nM T02001 CC1LZ4 24774931 IC50 = 160 nM T02001 CD9HX3 24774932 IC50 = 28 nM T02001 CVM84E 24775012 IC50 = 23 nM T02001 CE4CZ8 24775016 IC50 = 40 nM T02001 CM36BF 24775103 IC50 = 120 nM T02001 COZW45 24775104 IC50 = 100 nM T02001 CBZ24N 24775188 IC50 = 40 nM T02001 CC2QP4 24775189 IC50 = 150 nM T02001 CQ19ZC 24775191 EC50 = 66900 nM T02001 C1ZUO8 24775388 IC50 = 44 nM T02001 CT0RS8 24775389 IC50 = 65 nM T02001 C1US5O 24775390 IC50 = 67 nM T02001 CF16AW 24775573 IC50 = 32 nM T02001 CPQ0B5 24775658 IC50 = 36 nM T02001 C76UCA 24775659 IC50 = 18 nM T02001 C9HLW6 24775661 IC50 = 44 nM T02001 CKNA60 24775662 IC50 = 21 nM T02001 CXOZ31 24775752 IC50 = 46 nM T02001 CS17UZ 24775939 IC50 = 90 nM T02001 CF62OT 24775940 IC50 = 70 nM T02001 C82YMG 24775941 IC50 = 30 nM T02001 CGS30K 24775942 IC50 = 130 nM T02001 CD08OZ 24775943 IC50 = 30 nM T02001 CT78AF 24776039 IC50 = 140 nM T02001 CGO3U4 24776040 IC50 = 60 nM T02001 CE29LR 24776042 IC50 = 20 nM T02001 CUEC50 24776128 IC50 = 40 nM T02001 CTF70M 24776131 IC50 = 130 nM T02001 CDC36W 24776132 IC50 = 100 nM T02001 C9WGI4 24802717 IC50 = 5540 nM T02001 C20VHK 24871823 IC50 = 9610 nM T02001 C17XKA 24957745 IC50 = 20 nM T02001 CC9EB2 24957749 IC50 = 81 nM T02001 CR4A6X 24959218 IC50 = 63 nM T02001 COK7S0 24959219 IC50 = 15 nM T02001 C7T3AY 24959954 IC50 = 45 nM T02001 C6EQG2 24963293 IC50 > 2000 nM T02001 C42AKZ 25120500 IC50 = 0.5 nM T02001 C4YT9V 25147797 IC50 = 21.88 nM T02001 C93DZI 25147798 IC50 = 18.2 nM T02001 CC3M2K 25178110 IC50 = 10000 nM T02001 CR16QH 25178733 IC50 = 93325.43 nM T02001 C6BWC9 25178734 IC50 = 29000 nM T02001 CS17JC 25178735 IC50 = 60000 nM T02001 CY8J7K 25178736 IC50 = 70794.58 nM T02001 CF1RU9 25178737 IC50 = 23988.33 nM T02001 CQL8C0 25178738 IC50 = 100000 nM T02001 CP41KJ 25178916 IC50 = 102000 nM T02001 C1O7TS 25178917 IC50 = 44668.36 nM T02001 CS3W8X 25178918 IC50 = 724.44 nM T02001 CE9K1W 25178919 IC50 = 199.53 nM T02001 C8ZD0X 25178920 IC50 = 430 nM T02001 CRM69O 25178921 IC50 = 2290.87 nM T02001 C3B9ID 25178922 IC50 = 1900 nM T02001 C1GZ8X 25178923 IC50 = 2570.4 nM T02001 CJ28FP 25179109 IC50 = 407.38 nM T02001 CKWY57 25179110 IC50 = 177.83 nM T02001 C3SG2C 25179111 IC50 = 1096.48 nM T02001 CA29CE 25179112 IC50 = 180 nM T02001 C1PF8Q 25179114 IC50 = 2200 nM T02001 CRV0E8 25179115 IC50 = 39810.72 nM T02001 CMJ40D 25179281 IC50 = 5200 nM T02001 C7N1DI 25179284 IC50 = 10000 nM T02001 CPC08B 25179287 IC50 = 6000 nM T02001 CTK06Q 25179476 IC50 = 2570.4 nM T02001 CN65DU 25179477 IC50 = 380 nM T02001 COB03R 25179478 IC50 = 6000 nM T02001 C8YV0H 25179675 IC50 = 61 nM T02001 CNZM75 25179676 IC50 = 667 nM T02001 CQ6M3L 25179677 IC50 = 636 nM T02001 CWC1O2 25179678 IC50 = 346.74 nM T02001 C89JPH 25179679 IC50 = 44000 nM T02001 CGC01Z 25179875 IC50 = 501.19 nM T02001 C4BZW2 25180832 IC50 = 1513561.25 nM T02001 C4X8WU 25181020 IC50 = 537031.8 nM T02001 CRT0O1 25181021 IC50 = 524807.46 nM T02001 C8P6WY 25181022 IC50 > 100000 nM T02001 CF6AD3 25211583 IC50 = 253 nM T02001 CVU7J1 25211682 IC50 = 106 nM T02001 CX07CK 25258806 IC50 = 2 nM T02001 CTQI51 26273258 IC50 = 49300 nM T02001 CN4W2U 27659581 IC50 = 88300 nM T02001 C6GQR8 30515311 IC50 = 22 nM T02001 C5Q0IN 42647289 IC50 = 2.1 nM T02001 CNIE98 44143458 IC50 = 1.9 nM T02001 C2SLH8 44324331 IC50 = 10 nM T02001 C8PNR4 44329482 IC50 > 100000 nM T02001 CUFO76 44329511 IC50 = 700 nM T02001 CA1R5M 44329613 IC50 = 540 nM T02001 CHR0G3 44329633 IC50 > 100000 nM T02001 CT3M4H 44329639 IC50 = 850 nM T02001 CXUC09 44329640 IC50 = 230 nM T02001 CA5MY8 44329642 IC50 = 300 nM T02001 CSD45M 44329651 IC50 = 90 nM T02001 CUA7P5 44329666 IC50 = 140 nM T02001 C26ZAE 44329668 IC50 = 1200 nM T02001 C1T7JL 44329669 IC50 = 2000 nM T02001 C2M3QE 44329683 IC50 = 130 nM T02001 C9R0OI 44329684 IC50 = 8500 nM T02001 CWM23U 44329685 IC50 > 100000 nM T02001 CQ2WU3 44329686 IC50 = 60 nM T02001 CMF1J2 44329702 IC50 = 1200 nM T02001 C5YO6L 44329893 IC50 = 3000 nM T02001 CT1C4U 44329894 IC50 = 800 nM T02001 C13HPW 44393651 IC50 = 15700 nM T02001 CJ6GB5 44393709 IC50 = 690 nM T02001 CE8TU4 44393929 IC50 = 79000 nM T02001 C8U2DW 44393934 IC50 = 30000 nM T02001 CQP01D 44393950 IC50 = 58250 nM T02001 C6A7JK 44393959 IC50 > 101000 nM T02001 CU1CQ8 44394047 IC50 = 1020 nM T02001 CTX1E5 44394060 IC50 = 95500 nM T02001 CLMW27 44405467 IC50 = 0.6 nM T02001 CR05OY 44405507 IC50 = 2.5 nM T02001 C7OA9V 44405510 IC50 = 0.5 nM T02001 CFY36C 44410864 IC50 = 2.3 nM T02001 CT1JW4 44410870 IC50 = 0.1 nM T02001 C3EI4T 44410882 IC50 = 74 nM T02001 C7NKA2 44410914 IC50 = 10 nM T02001 CGA5J0 44541350 IC50 = 670 nM T02001 CZM1R4 44541481 IC50 = 5910 nM T02001 C4C9RI 44541606 Ki = 1550 nM T02001 C2YC8S 44541610 IC50 = 4270 nM T02001 C7VT1G 44541743 IC50 = 3480 nM T02001 CJD73U 44565305 Ki = 1.2 nM T02001 CYR1J4 44588185 IC50 = 79432.82 nM T02001 C3L8AY 44588256 IC50 = 199.53 nM T02001 CBL2J9 45263650 IC50 > 10000 nM T02001 CX5Q1U 45484316 IC50 = 31622.78 nM T02001 CO1NT8 45484317 IC50 = 2511.89 nM T02001 CG03XH 45484327 IC50 = 6309.57 nM T02001 CG1S6M 45484341 IC50 = 398.11 nM T02001 C19WRQ 45484346 IC50 = 2511.89 nM T02001 CT53FB 45484347 IC50 = 1584.89 nM T02001 C36XLQ 46209046 IC50 > 10000 nM T02001 C2Q4YT 46209162 IC50 > 10000 nM T02001 CJOE41 46209386 IC50 > 10000 nM T02001 CV6R4I 46227215 IC50 = 0.3 nM T02001 CE0W4J 46227268 IC50 = 45 nM T02001 CY5FD9 46227269 IC50 = 23 nM T02001 CGEF56 46227285 IC50 = 14.3 nM T02001 C6YVM2 46227286 IC50 = 5.2 nM T02001 CU1J6V 46227291 IC50 = 0.4 nM T02001 CV13MB 46227305 IC50 = 45.9 nM T02001 COID57 46227306 IC50 = 16.4 nM T02001 CCP5O4 46227309 IC50 = 4.3 nM T02001 CV1N2M 46227326 IC50 = 2 nM T02001 CCI3U1 46227327 IC50 = 9.7 nM T02001 C0F9VM 46227328 IC50 = 1 nM T02001 CN1C2D 46231449 IC50 = 32 nM T02001 C7LEU4 46231450 IC50 = 47 nM T02001 CN6K1Z 46231506 IC50 = 83 nM T02001 C71YOW 46231609 IC50 = 39 nM T02001 C0KNQ5 46231671 IC50 = 54 nM T02001 C2V3ZJ 46232011 IC50 = 70 nM T02001 C7VCA5 46232194 IC50 = 37 nM T02001 C3PA8E 46232320 IC50 = 32 nM T02001 C1JOF3 46830337 Ki = 8370 nM T02001 C3RJL6 46830338 Ki = 147 nM T02001 C1YXQ7 46884033 Ki = 59000 nM T02001 CR75HO 46884094 Ki = 54400 nM T02001 C6TW3L 46884095 Ki = 17500 nM T02001 C7GJO6 46884096 Ki = 14200 nM T02001 C8DW2I 46884097 Ki = 83000 nM T02001 CGW26E 46884133 Ki = 3350 nM T02001 CZ2V3A 46884134 Ki = 2400 nM T02001 C8HJV2 46884135 Ki > 100000 nM T02001 CE8SV7 46884136 Ki > 100000 nM T02001 CK7PD2 46884170 Ki = 61000 nM T02001 CR5AU2 46884171 Ki = 22200 nM T02001 CHBX41 46884172 Ki = 65000 nM T02001 C9B0QC 46884216 Ki = 19000 nM T02001 CT1U9Q 46884217 Ki = 18000 nM T02001 CSDA49 46884218 Ki > 100000 nM T02001 CZ9T7B 46884219 Ki = 80900 nM T02001 C35KWX 46884255 Ki > 100000 nM T02001 CW8EK3 46884256 Ki > 100000 nM T02001 C67OIK 46884257 Ki > 100000 nM T02001 CJ36UA 46884298 Ki = 15300 nM T02001 CW1L6Q 46884299 Ki = 11500 nM T02001 CHF10C 46884300 Ki > 100000 nM T02001 C8I2CM 46884366 Ki = 48600 nM T02001 CVM1Q7 46884367 Ki = 12700 nM T02001 CPT67V 46884368 Ki = 51200 nM T02001 C0L7JC 46884416 Ki = 4440 nM T02001 CF0PI3 46915888 IC50 = 1.8 nM T02001 C3P2IN 46933992 IC50 = 0.6 nM T02001 CB2HS9 46933993 IC50 = 0.2 nM T02001 CZ7C3F 46933994 IC50 = 0.8 nM T02001 CQ5NF4 49780548 IC50 = 4.2 nM T02001 C9H4BC 49780549 IC50 = 119 nM T02001 C0EH7V 49865602 IC50 = 22.2 nM T02001 C89UPD 49865603 IC50 = 17 nM T02001 CV81PG 49865604 IC50 = 10.5 nM T02001 C43XGJ 49865605 IC50 = 4.5 nM T02001 CIT05Z 49865642 IC50 = 18.3 nM T02001 C5OI1V 49865643 IC50 = 0.9 nM T02001 C19JZB 49866243 IC50 = 9.3 nM T02001 CU5B8G 49866268 IC50 = 0.4 nM T02001 CSYL46 49866269 IC50 = 5 nM T02001 CI3F7K 49866270 IC50 = 12.1 nM T02001 C7V8DY 49866271 IC50 = 48.7 nM T02001 CCJ7I1 49866272 IC50 = 2 nM T02001 C6R4YN 50993785 IC50 = 10000 nM T02001 C0M6XL 50993786 IC50 = 10000 nM T02001 CC36QO 53393812 IC50 = 290 nM T02001 CC18WN 54579989 IC50 = 7600 nM T02001 CZM4S8 54579990 IC50 = 82 nM T02001 CDR9V3 54580135 IC50 = 11000 nM T02001 CX1LD8 54581119 IC50 = 3000 nM T02001 C9H8CS 54581120 IC50 = 1300 nM T02001 C2RD7T 54583103 IC50 = 8800 nM T02001 C3YD5S 54583104 IC50 = 760 nM T02001 CS0A2F 54583105 IC50 = 2900 nM T02001 CP1ZD8 54583972 IC50 = 3400 nM T02001 CJ5ZV7 54584101 IC50 = 9900 nM T02001 CF3HA7 54585042 IC50 = 1300 nM T02001 C3-FEB-08 54585043 IC50 = 12000 nM T02001 CG54MF 54585044 IC50 = 5300 nM T02001 CAI3B7 54585882 IC50 = 2100 nM T02001 CBF2W8 54586013 IC50 = 2400 nM T02001 CYI6K8 54586014 IC50 > 10000 nM T02001 C38ZLC 54586015 IC50 = 4800 nM T02001 CT1A3P 54586846 IC50 = 1500 nM T02001 CK6QW0 54586848 IC50 = 1500 nM T02001 C2FN8X 54586849 IC50 = 8000 nM T02001 C8IO0C 54586990 IC50 = 15000 nM T02001 C3L9NI 54586991 IC50 = 2800 nM T02001 C52NHY 54586992 IC50 = 1500 nM T02001 C5DO4H 54586993 IC50 = 2000 nM T02001 CXR9T5 54586994 IC50 = 1500 nM T02001 CFX89L 54587804 IC50 = 2200 nM T02001 CLH72B 54591641 IC50 = 150 nM T02001 CGF65A 54670110 IC50 > 30000 nM T02001 C90ZLC 54670399 IC50 = 581 nM T02001 CK0Q2T 54764160 IC50 = 27 nM T02001 CHT86A 56642417 IC50 = 9.4 nM T02001 CBV60W 56642529 IC50 = 2.3 nM T02001 CKGD94 56642530 IC50 = 13.5 nM T02001 CKTD52 56642531 IC50 = 2.7 nM T02001 C4G6TL 56642532 IC50 = 14 nM T02001 CRK35Q 56642533 IC50 = 1.5 nM T02001 CF7P1Y 56642534 IC50 = 17 nM T02001 CP9CD7 56642658 IC50 = 240 nM T02001 CM8U9E 56642659 IC50 = 1.3 nM T02001 CAN50G 56642660 IC50 = 0.5 nM T02001 CPC3T4 56654131 IC50 > 10000 nM T02001 C1AND4 56659469 IC50 = 17 nM T02001 CGWH19 56662928 IC50 = 32 nM T02001 CQT17K 56662929 IC50 = 0.51 nM T02001 CLMG01 56662930 IC50 = 0.52 nM T02001 CL1U3W 56666405 IC50 = 0.66 nM T02001 C5H9XA 56669821 IC50 = 0.55 nM T02001 CIX9M0 56673307 IC50 = 0.46 nM T02001 CTY48D 56673902 IC50 = 4.6 nM T02001 CEO42M 56676640 IC50 = 0.58 nM T02001 C2CRW3 56679969 IC50 = 1 nM T02001 CT8A6K 56683302 IC50 = 0.35 nM T02001 CB17SC 57385767 IC50 = 66300 nM T02001 C59YAC 57495353 IC50 = 4700 nM T02001 CC6E2M 57703712 IC50 = 27 nM T02001 C4XMB6 58547809 IC50 > 30000 nM T02001 CEB3G9 58547814 IC50 = 5050 nM T02001 C08QVG 58547833 IC50 = 10800 nM T02001 CFVG67 58547863 IC50 = 4690 nM T02001 CYZA38 58548077 IC50 = 20500 nM T02001 CLEA86 59187022 IC50 = 3760 nM T02001 CW24YS 59190451 IC50 = 0.01995 nM T02001 CEI8A5 59190544 IC50 = 0.01995 nM T02001 CWX3N7 59320301 IC50 = 2060 nM T02001 C0EP5I 59341847 IC50 = 2500 nM T02001 CHQ28A 59341978 IC50 = 2120 nM T02001 CJ0YB8 59351288 IC50 > 10000 nM T02001 CCA1H6 59351376 IC50 > 10000 nM T02001 CM56CF 66829650 IC50 = 17 nM T02001 CA76CF 66829675 IC50 = 1 nM T02001 CVKU30 66829804 IC50 = 13 nM T02001 CU49WI 66829828 IC50 = 3 nM T02001 CUG2M9 66881198 IC50 = 13 nM T02001 C4HBV7 67030924 IC50 = 61 nM T02001 CW1ZP6 67030970 IC50 = 5 nM T02001 C6D5CB 67031033 IC50 = 212 nM T02001 CY8J3O 68181896 IC50 > 30000 nM T02001 CTEM06 68957324 IC50 > 10000 nM T02001 CN4DR0 69619707 Ki = 0.2344 nM T02001 COI2P3 70679302 IC50 > 10000 nM T02001 C2HGI7 71153408 IC50 > 10000 nM T02001 C0O6TB 71254628 IC50 = 1.8 nM T02001 CWF39E 71254723 IC50 = 1500 nM T02001 C93LAB 71254931 IC50 = 6.6 nM T02001 CF90QO 71262535 IC50 = 150 nM T02001 C14TJO 71262536 IC50 = 2300 nM T02001 C7AQH0 71262640 IC50 = 5.5 nM T02001 CU7DZ1 71262641 IC50 = 18 nM T02001 CR5NQ6 71450591 IC50 > 10000 nM T02001 CGD56M 71450592 IC50 > 10000 nM T02001 CJ62MK 71451776 IC50 = 31 nM T02001 C2UK6B 71451779 IC50 = 74 nM T02001 CZ1YN2 71452430 IC50 > 10000 nM T02001 CI1M8Q 71452431 IC50 > 10000 nM T02001 CX5D2O 71454197 IC50 > 10000 nM T02001 CJV1G2 71455939 IC50 > 10000 nM T02001 C8A4ME 71457746 IC50 > 10000 nM T02001 C6PS5B 71458967 IC50 = 140 nM T02001 C3VKH8 71459650 IC50 > 10000 nM T02001 CJ3Z7K 71460703 IC50 = 1.2 nM T02001 CT2D6E 71461384 IC50 = 7400 nM T02001 CHD9Q2 71512292 IC50 = 32 nM T02001 CNZ3L1 71552789 IC50 = 650 nM T02001 CYZS90 71552873 IC50 = 2890 nM T02001 C0WZ3P 71624963 IC50 = 1300 nM T02001 C6SP8E 71624964 IC50 = 550 nM T02001 C3HMB0 71625351 IC50 = 180 nM T02001 C68SDB 71719394 IC50 = 0.631 nM T02001 CUJ15C 71719800 IC50 = 3330 nM T02001 CZ0G2X 72165213 IC50 > 10000 nM T02001 C7XRY6 72190879 IC50 = 14882 nM T02001 CBM61I 73293715 IC50 = 2230 nM T02001 CHR7D0 73334611 IC50 = 13500 nM T02001 C9ODB8 73387740 IC50 = 8920 nM T02001 C5X6GJ 73387742 IC50 > 20000 nM T02001 CT1E6V 73387743 IC50 = 9540 nM T02001 C7D1SJ 73387744 IC50 = 14200 nM T02001 CG89ET 73387745 IC50 > 20000 nM T02001 C3HSE2 73387863 IC50 > 20000 nM T02001 C3R0TC 73387959 IC50 = 4270 nM T02001 CHFG14 73425856 IC50 = 4220 nM T02001 C74TSX 73425972 IC50 = 1780 nM T02001 CWX3M6 73425973 IC50 = 7850 nM T02001 CEH2R6 73425974 IC50 = 2980 nM T02001 CK5SA7 73425975 IC50 = 4270 nM T02001 CD3BZ0 73603954 IC50 = 219 nM T02001 CLR80D 74221042 IC50 = 3580 nM T02001 CCZ1V0 74221043 IC50 = 886 nM T02001 C7Y2JO 74221099 IC50 = 865 nM T02001 CBM14E 74221100 IC50 = 207 nM T02001 CQ2KG4 74221101 IC50 = 251 nM T02001 C8D4KG 74221105 IC50 = 1489 nM T02001 CC37TX 74221165 IC50 = 1181 nM T02001 C64ZJD 74221166 IC50 = 5611 nM T02001 CUTB06 74221167 IC50 = 268 nM T02001 C7IYQ1 74221168 IC50 = 681 nM T02001 CSP7M5 74221169 IC50 = 213 nM T02001 C3CSM1 74221170 IC50 = 2268 nM T02001 CLG7T8 74221229 IC50 = 20 nM T02001 CAUC08 74221233 IC50 = 2107 nM T02001 CB9GN2 74221235 IC50 = 268 nM T02001 C1QRG0 74221297 IC50 = 7 nM T02001 C6V1FJ 74221298 IC50 = 13 nM T02001 CX5H8N 74221299 IC50 = 132 nM T02001 CTU9V5 74221300 IC50 = 63 nM T02001 C04QOM 74221361 IC50 = 96 nM T02001 CKBM41 74221363 IC50 = 600 nM T02001 C9JE6M 75815419 IC50 = 26.3 nM T02001 CLGM26 76283410 IC50 = 200 nM T02001 CYZ02X 76283663 IC50 = 90 nM T02001 CCVE67 76283664 IC50 = 10 nM T02001 C1LCQ5 76310584 IC50 = 1300 nM T02001 CNY85L 76310585 IC50 = 290 nM T02001 CGN2F0 76310586 IC50 = 440 nM T02001 CS4GB6 76310587 IC50 = 1300 nM T02001 CZWC27 76314221 IC50 = 1800 nM T02001 CLXO82 76314222 IC50 = 2200 nM T02001 CHKB59 76314223 IC50 = 2100 nM T02001 CHC31S 76314224 IC50 = 3800 nM T02001 CYC23W 76314225 IC50 = 1000 nM T02001 C1X5GR 76314226 IC50 = 1300 nM T02001 CDWE89 76317790 IC50 = 1000 nM T02001 CFQ0P3 76317791 IC50 = 420 nM T02001 CPBL42 76317792 IC50 = 1600 nM T02001 CWB80L 76317793 IC50 = 400 nM T02001 C4KH2T 76321500 IC50 = 3400 nM T02001 C1XTZ7 76321501 IC50 = 860 nM T02001 C34RGJ 76321502 IC50 = 1100 nM T02001 C1TS0Y 76321503 IC50 = 580 nM T02001 C93VYC 76321504 IC50 = 560 nM T02001 CENO19 76321505 IC50 = 600 nM T02001 C78QEP 76325104 IC50 = 680 nM T02001 CSMV71 76325105 IC50 = 280 nM T02001 CNBJ29 76325106 IC50 = 3400 nM T02001 C5P9TA 76325107 IC50 = 620 nM T02001 CO8J5I 76328668 IC50 = 1000 nM T02001 CP1T2G 76328669 IC50 = 430 nM T02001 CH5Z2P 76328670 IC50 = 520 nM T02001 CWM15I 76328671 IC50 = 1300 nM T02001 CFA85S 76328672 IC50 = 810 nM T02001 C1A4WZ 76332343 IC50 = 300 nM T02001 C6R2XP 76332344 IC50 = 290 nM T02001 CW4Y7O 76332345 IC50 = 790 nM T02001 C2J6IZ 76332346 IC50 = 7400 nM T02001 CTXG71 76332347 IC50 = 1500 nM T02001 CCFA47 76332348 IC50 = 1200 nM T02001 CWKO07 76335973 IC50 = 790 nM T02001 CL3D1Y 76335974 IC50 = 1300 nM T02001 CB64TA 76335975 IC50 = 600 nM T02001 CXA0Y3 76335976 IC50 = 1400 nM T02001 CLW8D4 77461017 IC50 = 8 nM T02001 C8BO3W 90113029 IC50 = 22260 nM T02001 CG5P9A 90153688 IC50 = 4200 nM T02001 CUR62C 90154140 IC50 = 4500 nM T02001 CN85IK 90655366 IC50 = 16650 nM T02001 C5NXL4 90655367 IC50 = 7810 nM T02001 CGO6Y3 90655368 IC50 = 140 nM T02001 CA62ZP 90655369 IC50 = 1530 nM T02001 C2CFZ5 90655370 IC50 = 11490 nM T02001 CY3IW6 90655371 IC50 = 10220 nM T02001 C4RN9B 90667924 IC50 = 2840 nM T02001 C1JPD6 91844700 IC50 = 4000 nM T02001 C4F7UM 92471957 IC50 = 250 nM T02001 CYQV05 92471958 IC50 = 5.4 nM T02001 C9VBM1 101784404 IC50 = 13273 nM T02001 C79YRO 101784407 IC50 > 20000 nM T02001 C9AQF2 101815805 IC50 = 4700 nM T02001 CQCA74 101886683 IC50 = 3000 nM T02001 CG3ZT2 102584765 IC50 = 5500 nM T02001 CECS24 102584766 IC50 = 1400 nM T02001 CHY06X 102584767 IC50 = 3700 nM T02001 CQ9PN8 102593934 IC50 = 6600 nM T02001 CSCY01 117949009 IC50 > 10000 nM T02001 C21HKZ 118048422 IC50 = 160 nM T02001 CNX7M9 118473558 IC50 = 10400 nM T02001 CYQ74R 118479645 IC50 > 10000 nM T02001 C8CM1B 118707986 IC50 = 3790 nM T02001 CK7E8J 118707987 IC50 = 2010 nM T02001 C6Y3WJ 118707988 IC50 = 8 nM T02001 CBP20D 118707989 IC50 = 11 nM T02001 CC6B5L 118707990 IC50 = 17 nM T02001 CW7TU1 118708069 IC50 = 727 nM T02001 CE59WQ 118708071 IC50 = 859 nM T02001 C6VT7X 118708072 IC50 = 726 nM T02001 CR7YV2 118711351 IC50 = 1550 nM T02001 C7PQT4 118711355 IC50 = 1790 nM T02001 CLE68Z 118711357 IC50 = 1260 nM T02001 C2S9TF 118711358 IC50 = 210 nM T02001 CR75BH 118712216 IC50 = 7.3 nM T02001 CJIY54 118712217 IC50 = 48 nM T02001 C0NQ6I 118712218 IC50 = 7200 nM T02001 C3XM4A 118712219 IC50 > 10000 nM T02001 C6KRJ9 118712220 IC50 = 9.9 nM T02001 C86PHO 118712221 IC50 = 4.5 nM T02001 CD82CM 118712222 IC50 = 170 nM T02001 CI84UJ 118713845 IC50 = 10600 nM T02001 CDF95E 118713849 IC50 = 12100 nM T02001 C5TK4E 118713851 IC50 = 16900 nM T02001 C42AZD 118713853 IC50 = 7200 nM T02001 C4FYN8 118713854 IC50 = 5900 nM T02001 C2B4AK 118713855 IC50 = 3600 nM T02001 CG0AB1 118716213 IC50 > 20000 nM T02001 CT9H7V 121285043 IC50 = 9200 nM T02001 C1XNB3 122179937 IC50 = 1490 nM T02001 C08ONI 122179938 IC50 = 190 nM T02001 CZUI96 122179939 IC50 = 2540 nM T02001 CX12NJ 122179940 IC50 = 190 nM T02001 CH2OT7 122179941 IC50 = 1120 nM T02001 C1D0EJ 122179942 IC50 = 4840 nM T02001 C6RBJ7 122179943 IC50 = 2630 nM T02001 CJ0C7S 122179944 IC50 = 470 nM T02001 CRJE23 122185011 IC50 = 7620 nM T02001 CS80MH 122193673 IC50 = 284 nM T02001 C8CJU5 122193675 IC50 = 342 nM T02001 CS6M9C 122193679 IC50 = 94 nM T02001 CQV4W1 122193754 IC50 = 108 nM T02001 C4PLA1 124525843 IC50 = 2190 nM T02001 C90DLV 127025000 IC50 = 542 nM T02001 CVX7U9 127029185 IC50 = 245 nM T02001 CI50YP 127033692 IC50 = 486 nM T02001 C6AC9Z 127033706 IC50 = 3100 nM T02001 COI63Z 127033976 IC50 = 6070 nM T02001 C3QN7O 127034775 IC50 = 3050 nM T02001 C9ZR8J 127034776 IC50 = 2080 nM T02001 CW95MQ 127034954 IC50 = 2920 nM T02001 CVBL45 127034956 IC50 = 320 nM T02001 CGZ85U 127035574 IC50 > 10000 nM T02001 CAY68J 127035760 IC50 = 3670 nM T02001 CN8O4U 127035761 IC50 = 750 nM T02001 C3Y2WC 127037266 IC50 = 2310 nM T02001 C92BNQ 127037472 IC50 = 960 nM T02001 CAE14X 127053189 IC50 > 20000 nM T02001 C9AGC4 127053190 IC50 > 20000 nM T02001 CD5NK3 127053211 IC50 > 20000 nM T02001 CS4JD0 129626433 IC50 = 62 nM T02001 CW2HR1 130366728 IC50 = 306 nM T02001 C2ALN7 130366739 IC50 > 15100 nM T02001 CQJN83 130366758 IC50 > 29800 nM T02001 CDAF16 130380472 IC50 > 12800 nM T02001 C18KLO 130380505 IC50 > 12200 nM T02001 C5XCO1 130380512 IC50 = 558 nM T02001 CT2E8Q 130380575 IC50 = 6420 nM T02001 CACJ46 132489333 IC50 = 2769 nM T02001 CG8HF1 132938287 IC50 = 10600 nM T02001 C2P1IU 134129996 IC50 = 22 nM T02001 CLE03O 134130328 IC50 = 68 nM T02001 CSN6J0 134130563 IC50 = 71 nM T02001 C0A1CZ 134131162 IC50 = 39 nM T02001 C1GY2T 135156251 EC50 > 10000 nM T02001 C3R8SE 135457869 IC50 > 10000 nM T02001 CJS37E 135482260 IC50 = 820 nM T02001 C1RK8U 135815296 Ki = 4.1 nM T02001 C3PO9K 135856789 IC50 = 5630 nM T02001 C3M7VF 135856791 IC50 = 12230 nM T02001 CAO3U7 135856794 IC50 = 71000 nM T02001 CTX54Z 135896326 IC50 > 10000 nM T02001 CIW37T 136035260 IC50 = 650 nM T02001 C12UMG 136059728 IC50 > 1000 nM T02001 C2VO1H 136132220 Ki = 3.7 nM T02001 C8PG9Q 136132221 Ki = 5.1 nM T02001 CUI4W9 136132222 Ki = 3 nM T02001 CST26Q 136132223 Ki = 7.4 nM T02001 CQ27TM 136132224 Ki = 590 nM T02001 CMIY85 136132225 Ki = 4.9 nM T02001 C7J3IT 136132226 Ki = 7.8 nM T02001 CT3IC8 136132227 Ki = 322 nM T02001 CYM29K 136132228 Ki = 5.1 nM T02001 CEM5N1 136132229 Ki = 4300 nM T02001 C4V5AD 136132230 Ki = 7.9 nM T02001 CJC0X9 136132231 Ki = 114.7 nM T02001 COA9T2 136132232 Ki = 5.6 nM T02001 CQ50CG 136132233 Ki = 9.9 nM T02001 CY50JV 136132234 Ki = 6.6 nM T02001 C28IYL 136132235 Ki = 13 nM T02001 CHW75A 136132236 Ki = 6.6 nM T02001 C9GA2W 136132237 Ki = 19.4 nM T02001 C39MDZ 136132238 Ki = 4.3 nM T02001 CW3FM6 136132239 Ki = 4.8 nM T02001 C5XBZ6 136132240 Ki = 6.3 nM T02001 CU8RC1 136132241 Ki = 6.5 nM T02001 C5NVZ9 136132242 Ki = 6.8 nM T02001 CF31SZ 136132243 Ki = 6.6 nM T02001 C8TQ7A 136217455 IC50 = 15700 nM T02001 CE4HQ5 136230157 IC50 = 6550 nM T02001 CI1W8Q 136230159 IC50 = 2900 nM T02001 CY8PZ4 137175273 IC50 = 8860 nM T02001 CKD31C 137175274 IC50 = 2010 nM T02001 C3BM9A 137175275 IC50 = 1070 nM T02001 C81PHA 137189790 IC50 = 890 nM T02001 CD8ZA9 137189803 IC50 = 230 nM T02001 C4KZA9 137189822 IC50 > 10000 nM T02001 C6XG1B 137189823 IC50 = 1210 nM T02001 C2N9VT 137348687 IC50 > 10000 nM T02001 CUX5J6 137628440 IC50 = 33800 nM T02001 C26WMG 137628497 IC50 = 5400 nM T02001 C59ABT 137628530 IC50 = 2800 nM T02001 C3GT9X 137628532 IC50 = 29500 nM T02001 CFVS01 137628547 IC50 = 1200 nM T02001 C12FGT 137628551 IC50 = 19500 nM T02001 CT64GE 137628564 IC50 = 23200 nM T02001 CAB1M3 137628580 IC50 = 24600 nM T02001 CCB4A5 137628587 IC50 = 32100 nM T02001 C9P3UR 137637125 IC50 = 31650 nM T02001 C92JAF 137637269 IC50 = 12830 nM T02001 CYJ75P 137640039 IC50 = 23120 nM T02001 CH7QG9 137645629 IC50 = 8400 nM T02001 CYK2A9 137646728 IC50 = 13880 nM T02001 COGR93 137649084 IC50 = 23320 nM T02001 C2TZM4 137650925 IC50 = 5130 nM T02001 CE69UN 137651372 IC50 = 7150 nM T02001 CLN2U7 137652270 IC50 = 700 nM T02001 CXS6E7 137658977 IC50 = 1600 nM T02001 CA4J9M 137662320 IC50 = 26750 nM T02001 C6KYD7 137700754 IC50 > 10000 nM T02001 CF2VM7 137700766 Ki = 0.123 nM T02001 CKA14E 137700767 Ki = 0.3548 nM T02001 C0N6LV 137700768 Ki = 0.1549 nM T02001 CSDP84 137700769 Ki = 0.302 nM T02001 CM3UF7 137700779 IC50 > 20000 nM T02001 CPTE92 138319693 IC50 = 43 nM T02001 C2QLX3 138393292 IC50 = 240 nM T02001 C5JG7H 139267726 IC50 = 20700 nM T02001 CKO4F5 139267727 IC50 = 26100 nM T02001 CJ16QH 139267728 IC50 = 650 nM T02001 CFUT09 139267729 IC50 = 4300 nM T02001 CU98MJ 139267730 IC50 = 250 nM T02001 CMX2Y1 139267731 IC50 = 270 nM T02001 CG0FQ5 139399269 IC50 = 98 nM T02001 C7BF2N 139399292 IC50 = 510 nM T02001 C4ZMA3 139399298 IC50 = 3710 nM T02001 CVAM65 139399322 IC50 = 820 nM T02001 CUN3G2 139399340 IC50 = 130 nM T02001 C87OQT 139399398 IC50 = 700 nM T02001 CQ3HB0 140943145 IC50 = 380 nM T02001 C1S7HV 142592633 IC50 = 385 nM T02001 CN3OC2 142592634 IC50 = 108 nM T02001 CY64NR 142592636 IC50 = 360 nM T02001 C83XNL 142592649 IC50 = 220 nM T02001 C7XZB1 142592652 IC50 = 136 nM T02001 CQG91H 145949384 IC50 = 4890 nM T02001 C2NR0Z 145949558 IC50 = 1880 nM T02001 C9SH7Y 145949856 IC50 > 30000 nM T02001 CV5G0Y 145949858 IC50 = 20 nM T02001 C0MT4D 145950945 IC50 = 25200 nM T02001 C81BLG 145951005 IC50 = 35000 nM T02001 C56ESR 145951756 IC50 = 30 nM T02001 C0BQ7T 145952944 IC50 = 50100 nM T02001 C0MO2L 145953102 IC50 = 89200 nM T02001 C3JY9H 145953411 IC50 = 15600 nM T02001 CW57KB 145953738 IC50 = 9210 nM T02001 CA2HD7 145955008 IC50 = 270 nM T02001 C9EC6O 145955031 IC50 = 40300 nM T02001 CBS1F9 145955232 IC50 = 10200 nM T02001 C5S9UB 145955505 IC50 = 8600 nM T02001 C1ES7U 145955804 IC50 = 9900 nM T02001 CL03PE 145955854 IC50 = 10300 nM T02001 CJYB46 145957166 IC50 = 870 nM T02001 CD5R3O 145957727 IC50 = 96800 nM T02001 CH3S7I 145958166 IC50 = 32000 nM T02001 CE6H8B 145958366 IC50 = 7500 nM T02001 C8LJ7Q 145958555 IC50 = 23000 nM T02001 CF6Q3V 145958985 IC50 = 5180 nM T02001 CRX30Z 145959784 IC50 = 56800 nM T02001 CWUZ70 145960159 IC50 = 81300 nM T02001 CYS17B 145965099 IC50 = 6500 nM T02001 CEGI75 145965101 IC50 = 5.07 nM T02001 CW6R4V 145965268 IC50 = 18270 nM T02001 CDYL80 145967203 IC50 = 2.73 nM T02001 C2XMK5 145972668 IC50 = 4350 nM T02001 CL46GW 145973062 IC50 = 43620 nM T02001 CFS8N5 145973376 IC50 = 18100 nM T02001 CZAJ58 145973921 IC50 = 32680 nM T02001 CC7HN2 145974174 IC50 = 18400 nM T02001 C9RGV1 145974955 IC50 = 16320 nM T02001 C2GIR6 145975414 IC50 = 133560 nM T02001 CP9R8Z 145976467 IC50 = 13260 nM T02001 C5NR0W 145976583 IC50 = 92580 nM T02001 C8MT9S 145977100 IC50 = 18620 nM T02001 CK1BR0 145978345 IC50 = 11650 nM T02001 CG0C4K 145978810 IC50 = 4.54 nM T02001 CG3M8I 145980160 IC50 > 100000 nM T02001 CM31VB 145980561 IC50 = 43 nM T02001 CD4I2X 145981417 IC50 = 18 nM T02001 CK7E5P 145981833 IC50 = 2400 nM T02001 CK45RB 145981967 IC50 = 52900 nM T02001 C4HJ5U 145983187 IC50 = 49300 nM T02001 C6K2MS 145987191 IC50 = 9600 nM T02001 C9TYX0 145987253 IC50 = 87300 nM T02001 CYP36H 145987360 IC50 = 13 nM T02001 CSN8W5 145987530 IC50 = 5600 nM T02001 CEA20L 145987749 IC50 = 15 nM T02001 C4A2KP 145987909 IC50 > 33000 nM T02001 C9CMG6 145989684 IC50 = 6 nM T02001 CB6MV7 145990536 IC50 = 88200 nM T02001 CL68MB 145990931 IC50 = 32 nM T02001 CZ37YN 145992861 IC50 = 24 nM T02001 CPD5L1 145993291 IC50 = 26400 nM T02001 C42OZA 145993939 IC50 = 19600 nM T02001 C35PRD 145994244 IC50 = 88 nM T02001 C8X2IT 145996536 IC50 = 210 nM T02001 CHJ79V 145997874 IC50 = 17 nM T02001 C6YG5B 149744413 IC50 = 99 nM T02001 CEZ2F8 150023808 IC50 = 16 nM T02001 CIG01L 150234338 IC50 = 44 nM T02001 CYR2X4 151339441 IC50 > 10000 nM T02001 C4FU1A 152008370 IC50 = 76 nM T02001 C0B4RN 152346644 IC50 = 480 nM T02001 CU1VK2 152504383 IC50 > 10000 nM T02001 CSL61Y 152626662 IC50 = 58 nM T02001 CCE9M0 153535392 IC50 > 10000 nM T02001 CU80DE 155510785 IC50 = 426 nM T02001 CHI38T 155511078 Ki = 0.1202 nM T02001 CR2M8W 155512088 IC50 > 10000 nM T02001 CEKJ30 155514856 IC50 > 10000 nM T02001 C46KSE 155514873 IC50 = 4640 nM T02001 CT1U8S 155515677 Ki = 0.1622 nM T02001 CT9W1I 155516764 IC50 = 22040 nM T02001 CBGL96 155516849 IC50 = 1077 nM T02001 C2MB4E 155517261 Ki = 0.3162 nM T02001 C7ADJ4 155517406 IC50 = 597 nM T02001 CX8VY5 155517795 IC50 = 1307 nM T02001 C03WPT 155518716 IC50 = 4930 nM T02001 CQ2IK7 155519106 IC50 = 399 nM T02001 C7JPT1 155519178 IC50 = 26160 nM T02001 COJ27G 155520087 IC50 = 622 nM T02001 C2ZCI9 155521531 IC50 > 10000 nM T02001 CL8CU6 155521936 IC50 = 6660 nM T02001 CDI7Z6 155521989 Ki = 63.1 nM T02001 C0ZV1F 155522911 Ki = 0.1549 nM T02001 CCXN80 155523172 Ki = 0.871 nM T02001 C1INP5 155523561 Ki = 0.5623 nM T02001 C8O7BF 155523628 IC50 = 87 nM T02001 COKA60 155523996 IC50 = 4600 nM T02001 C9GM2I 155524355 IC50 = 7360 nM T02001 CT91UI 155524447 IC50 > 10000 nM T02001 CX3Y7J 155525111 IC50 = 7630 nM T02001 C4YQZ5 155525638 IC50 = 5020 nM T02001 C0TK7O 155527643 IC50 = 8070 nM T02001 C1IT4X 155528561 Ki = 1.175 nM T02001 C0CGQ7 155528568 Ki = 0.1698 nM T02001 C4CL5F 155528672 Ki = 0.6761 nM T02001 CVG71O 155529178 IC50 = 6130 nM T02001 CW03OH 155529282 Ki = 30.2 nM T02001 C84KIS 155529462 IC50 > 10000 nM T02001 CV13TI 155529471 IC50 > 30000 nM T02001 CZQ39X 155530453 IC50 = 3830 nM T02001 CT85RG 155530589 IC50 = 5780 nM T02001 CK2U8G 155530765 Ki = 0.8511 nM T02001 C7NQU8 155531701 IC50 = 108 nM T02001 CC8M4K 155532035 Ki = 0.6607 nM T02001 C7PQT3 155532330 Ki = 2.57 nM T02001 CU7I9B 155532788 IC50 > 10000 nM T02001 CZ91HU 155533144 IC50 = 10690 nM T02001 CL3J5K 155533312 IC50 > 10000 nM T02001 C61PUD 155533540 IC50 = 934 nM T02001 CD26VI 155534361 IC50 = 4400 nM T02001 C4GQO3 155534561 IC50 = 15820 nM T02001 CNBI53 155535422 Ki = 0.6761 nM T02001 CK3U4A 155535738 Ki = 2.455 nM T02001 CQ30UY 155535906 IC50 = 32780 nM T02001 CWI0V6 155536272 Ki = 0.3162 nM T02001 C6JX9R 155537173 IC50 > 10000 nM T02001 CD4F2G 155537465 IC50 = 4150 nM T02001 CF7PQ6 155538533 IC50 = 7400 nM T02001 C42QIN 155539388 IC50 > 1000 nM T02001 CX62NF 155539572 IC50 = 99 nM T02001 CH2MO1 155543093 Ki = 0.5129 nM T02001 CFB3S9 155543476 IC50 = 271 nM T02001 CEMT29 155545548 IC50 = 38560 nM T02001 CM1T8W 155546720 Ki = 1.622 nM T02001 C7MW4U 155548627 IC50 = 148 nM T02001 CD6K2Y 155548709 IC50 = 29660 nM T02001 C6CJ2T 155548847 IC50 = 41 nM T02001 C8V4AW 155551577 IC50 = 37420 nM T02001 CK13EC 155552465 IC50 = 1071 nM T02001 CI5ZG4 155553883 IC50 = 25 nM T02001 CYBR26 155554299 IC50 = 501 nM T02001 CHI5G4 155554758 IC50 = 13700 nM T02001 C43BGO 155554947 IC50 > 10000 nM T02001 C3LQN9 155557352 IC50 = 3130 nM T02001 C3IC5U 155559413 IC50 = 200 nM T02001 CP2KO6 155560827 Ki = 2.455 nM T02001 CTL6O7 155562866 IC50 = 13780 nM T02001 C3CR6S 155563411 IC50 = 36680 nM T02001 C7KBJ3 155563967 IC50 = 11250 nM T02001 CR9V4W 155564375 IC50 = 477 nM T02001 CY4S1X 155564743 IC50 = 10130 nM T02001 C0CH3Y 155566295 IC50 = 15250 nM T02001 CAVX26 155567081 IC50 = 492 nM T02001 CTK08D 155567341 IC50 = 4060 nM T02001 C9AO6I 155567701 Ki = 0.2239 nM T02001 CI8WV3 155567794 IC50 = 11180 nM T02001 CD95BO 155568658 IC50 = 308 nM T02001 C2DY7M 155568806 Ki = 0.389 nM T02001 CJZ20G 155569371 IC50 = 6780 nM T02001 D00MBG 2921148 IC50 = 1280 nM T02001 D01RUN 448055 IC50 = 231 nM T02001 D01WTQ 5495929 IC50 = 420 nM T02001 D02FZD 158758 IC50 = 1000 nM T02001 D02NKD 10711281 IC50 = 2 nM T02001 D05UMA 10334821 IC50 > 100000 nM T02001 D06PRC 5281650 IC50 = 1310 nM T02001 D08AWN 3058751 IC50 >= 100000 nM T02001 D0I4TO 10107888 IC50 > 100000 nM T02001 D0JD4C 9853498 IC50 = 1.2 nM T02001 D0P2TS 9818682 IC50 = 900 nM T02001 D0R6MT 3758 IC50 = 31000 nM T02001 D0V4WB 149790 IC50 > 16000 nM T02001 D0W7WV 11039077 IC50 = 0.4 nM T02001 D0WB6P 46227262 IC50 > 100000 nM T02001 D0X7SR 10246505 IC50 = 630 nM T40954 D02ZXM 2723601 IC50 = 92420 nM T40954 D04AIT 5280445 IC50 = 550 nM T40954 D04KYY 135401907 IC50 = 1.6 ug.mL-1 T40954 D08IBS 190 IC50 = 10890 nM T40954 D0A5SE 134018 Ki = 0.1 nM T40954 D0E9CD 12127 IC50 > 50000 nM T40954 D0K8KX 5280343 Ki = 280 nM T40954 D0N0ES 938 IC50 = 518230 nM T40954 D04PBH 5280804 IC50 = 1600 nM T40954 D05TPI 72276 IC50 > 100000 nM T40954 D08FWK 135398752 Ki = 35 nM T40954 D0L4FS 5280961 IC50 = 232500 nM T40954 D07RPR 135413497 IC50 = 1000 nM T40954 D0E4FM 449035 IC50 = 5.8 nM T40954 C6ET5I 675 IC50 > 200000 nM T40954 CCJ6P5 4947 IC50 = 628000 nM T40954 C0NP3E 7195 IC50 = 86840 nM T40954 CAV1K2 7428 IC50 = 15520 nM T40954 CL9F3T 9955 IC50 > 200000 nM T40954 C8RI5S 11979 IC50 > 200000 nM T40954 CL70CJ 13650 IC50 = 131000 nM T40954 CG3Z6S 24667 IC50 = 591000 nM T40954 CZJ8U9 30976 IC50 > 200000 nM T40954 CVS6A8 40634 IC50 > 1000000 nM T40954 CW67XG 65275 IC50 > 200000 nM T40954 CL15AQ 65373 IC50 = 213000 nM T40954 CQ9MW6 68077 IC50 > 100000 nM T40954 C30ARD 70775 IC50 = 16700 nM T40954 CTK25Q 72277 IC50 > 100000 nM T40954 CJ65ZE 72344 IC50 > 100000 nM T40954 CPF12M 75420 IC50 = 30260 nM T40954 CKN0O5 92267 IC50 > 648000 nM T40954 CFT06L 127005 Ki > 100000 nM T40954 C8ZM5K 165506 IC50 > 30000 nM T40954 CK32ZP 176918 IC50 = 16800 nM T40954 C4IZP7 195123 IC50 = 97300 nM T40954 C1V0SM 219732 IC50 > 100000 nM T40954 CHW12S 220753 IC50 = 17350 nM T40954 CH13DO 221075 IC50 = 2200 nM T40954 C7PBC3 267626 IC50 = 31540 nM T40954 C3QV5H 287064 IC50 = 29640 nM T40954 CT43HC 326004 IC50 = 92 nM T40954 CT8D6X 385088 Ki = 2560 nM T40954 C7HME8 439246 IC50 > 50000 nM T40954 C5B4VP 639097 IC50 > 100000 nM T40954 CS04VD 641298 IC50 = 13.8 ug.mL-1 T40954 C2R3SD 772603 IC50 = 10000 nM T40954 C7XPG9 2179708 IC50 = 26100 nM T40954 CWU01F 2451195 IC50 = 36110 nM T40954 CA2T5J 2763873 IC50 > 100000 nM T40954 C6LM7G 2800424 IC50 > 100000 nM T40954 CIYF61 3004518 Ki > 100000 nM T40954 CQ21NS 4112136 Ki > 30000 nM T40954 CGI04J 5280536 IC50 = 36.3 ug.mL-1 T40954 C1BPI8 5280569 IC50 = 390000 nM T40954 CFP93L 5281603 IC50 = 36000 nM T40954 C65XQI 5281695 IC50 = 36500 nM T40954 C6KPO8 5281871 IC50 = 31500 nM T40954 CLN3V5 5282152 IC50 = 11900 nM T40954 C0WXP5 5284649 IC50 > 1000000 nM T40954 C4DUJ1 5315206 IC50 > 100000 nM T40954 C4H3EQ 5315892 IC50 > 50 ug.mL-1 T40954 CW31RM 5316262 IC50 = 101380 nM T40954 C97PDQ 5316728 IC50 > 50 ug.mL-1 T40954 CU0KV2 5317750 IC50 = 682600 nM T40954 C1I9ND 5318169 IC50 = 14.6 ug.mL-1 T40954 CW56EF 5318255 IC50 > 100000 nM T40954 CFG56S 5318767 IC50 = 14800 nM T40954 CRY76T 5319502 IC50 = 246000 nM T40954 CL6J0E 5320287 IC50 = 7700 nM T40954 CQP43H 5360349 IC50 > 200000 nM T40954 C1HZJ2 6438825 IC50 = 600 nM T40954 COG3B0 6440755 IC50 > 50 ug.mL-1 T40954 CHU87Y 10031889 IC50 = 6130 nM T40954 CJ2P6X 10036013 Ki = 1260 nM T40954 CL2KI8 10059496 Ki = 330 nM T40954 CW5B9D 10098455 IC50 = 94700 nM T40954 C30PGX 10101409 IC50 > 100000 nM T40954 C1LF5H 10258610 IC50 = 6520 nM T40954 CW4NA6 10325700 IC50 = 19500 nM T40954 C32EFC 10493305 IC50 = 36520 nM T40954 CH37BS 10563810 Ki = 1040 nM T40954 CSF45D 10564990 Ki = 93000 nM T40954 C59NKQ 10658574 Ki = 1060 nM T40954 C6RM3X 10776674 Ki = 2070 nM T40954 CTXL37 10802828 Ki = 260 nM T40954 C4GRI7 11168830 IC50 = 129000 nM T40954 C1U4SQ 11193310 IC50 = 178000 nM T40954 CUTV09 11758702 IC50 > 644000 nM T40954 CYHM16 11996550 IC50 = 400 nM T40954 CTW8N9 12952992 IC50 > 100000 nM T40954 CHJ9X7 13320505 IC50 > 100000 nM T40954 CP23SI 13991590 IC50 = 8260 nM T40954 CG3NM6 14642192 Ki = 40250 nM T40954 CR30KT 14642193 Ki = 66800 nM T40954 C2M5FK 15063047 Ki > 100000 nM T40954 CHP9N2 15063048 Ki = 24390 nM T40954 CUT36R 15063049 Ki = 131000 nM T40954 C2G6QS 24829407 IC50 = 80 nM T40954 CC48QW 24873793 IC50 > 100000 nM T40954 C9PA0D 24873794 IC50 = 37920 nM T40954 CKE50O 24873795 IC50 = 80970 nM T40954 CH3U2C 24873855 IC50 = 180 nM T40954 CKU03C 24873856 IC50 = 19580 nM T40954 C8GVB2 24873857 IC50 > 100000 nM T40954 CBC80Y 24873858 IC50 = 18440 nM T40954 CS5H2A 24896701 IC50 > 612000 nM T40954 CI3Q0K 24898465 IC50 = 42100 nM T40954 C9XED4 25147698 IC50 = 21300 nM T40954 CS24FX 25147699 IC50 = 131000 nM T40954 CMS03V 44178672 IC50 = 7710 nM T40954 C13IPT 44219681 IC50 = 96700 nM T40954 CQ6VW4 44326719 IC50 = 155750 nM T40954 C84CQX 44326901 IC50 = 139000 nM T40954 CHS56G 44326902 IC50 = 150000 nM T40954 C3Y9RP 44326903 IC50 = 102000 nM T40954 CWD2Z7 44326948 IC50 = 112000 nM T40954 CYAG83 44326949 IC50 = 129000 nM T40954 C7K8UC 44431346 IC50 = 21000 nM T40954 CN6B2U 44566544 IC50 > 100000 nM T40954 C3ET0R 44566545 IC50 > 100000 nM T40954 CDKJ28 44566578 IC50 = 150400 nM T40954 CP3U8V 44566579 IC50 = 79880 nM T40954 C5EKG9 44566586 IC50 = 110880 nM T40954 CS9CZ4 44575069 IC50 = 16000 nM T40954 CIQB14 44583918 Ki = 14350 nM T40954 C15OQK 44583919 IC50 > 100000 nM T40954 CZ5L0I 44593486 IC50 > 100000 nM T40954 CTX1E2 45266447 IC50 = 16500 nM T40954 C4I5ZE 45782989 IC50 > 100000 nM T40954 CCA01U 46881368 IC50 > 50 ug.mL-1 T40954 CL2O0Y 50994839 IC50 > 648000 nM T40954 C7OB2X 51035721 Ki > 30000 nM T40954 CB8ND9 51354813 IC50 > 679000 nM T40954 CCJ3R7 52915873 IC50 = 37800 nM T40954 CS8C9J 52915986 IC50 = 65500 nM T40954 CRK24I 52915987 IC50 = 47300 nM T40954 C1LW7J 52915988 IC50 = 108700 nM T40954 C4F5SK 52915989 IC50 = 56500 nM T40954 CH1KM7 52915990 IC50 = 82300 nM T40954 C89VMC 52915991 IC50 = 68800 nM T40954 C8BCL9 52915992 IC50 = 63000 nM T40954 C3H6ZO 52916097 IC50 = 72900 nM T40954 C8DNM4 52916098 IC50 = 53500 nM T40954 CWA9E7 52916099 IC50 = 91900 nM T40954 C7UA0N 52916100 IC50 = 44300 nM T40954 CFC42O 53323677 IC50 > 675000 nM T40954 CAS91K 54682930 IC50 = 195000 nM T40954 C5T8NI 56956282 IC50 = 15000 nM T40954 CY4WT8 57331330 IC50 = 4500 nM T40954 C4ALV1 57331603 IC50 = 4000 nM T40954 CLX5E7 57331685 IC50 = 5000 nM T40954 C3S7BJ 70692598 IC50 > 50 ug.mL-1 T40954 C3RK6L 70692599 IC50 > 50 ug.mL-1 T40954 CR9TD6 70694646 IC50 > 50 ug.mL-1 T40954 CXQ43R 71508608 IC50 = 49.4 nM T40954 CK13HD 71508609 IC50 = 24.5 nM T40954 C3E4LW 71508644 IC50 = 18.9 nM T40954 CQ2BV1 71508645 IC50 = 5.7 nM T40954 CUHL20 71508717 IC50 = 10.8 nM T40954 C7VJ1W 71539222 IC50 = 33.77 ug.mL-1 T40954 CZV2P3 71539941 IC50 = 77.74 ug.mL-1 T40954 CPR9J2 71539942 IC50 > 100 ug.mL-1 T40954 C4YKC7 71539982 IC50 = 34.1 ug.mL-1 T40954 CN91QB 71539983 IC50 = 38.79 ug.mL-1 T40954 C40QOC 71539984 IC50 > 100 ug.mL-1 T40954 CUE83P 71539985 IC50 = 89.28 ug.mL-1 T40954 CE83QY 71539986 IC50 = 61.25 ug.mL-1 T40954 C3RE7D 71539987 IC50 = 40.32 ug.mL-1 T40954 C1GRQ0 72375178 IC50 = 86.65 ug.mL-1 T40954 CSQF10 72375281 IC50 = 40.59 ug.mL-1 T40954 CM7F5W 72375282 IC50 = 36.83 ug.mL-1 T40954 C6Y8TR 76329670 IC50 = 1800 nM T40954 CG38DM 102429758 IC50 = 280 nM T40954 C0A3OH 118366073 IC50 = 37 nM T40954 C16VWC 118366086 IC50 = 29.3 nM T40954 CI27PO 118366091 IC50 = 35.2 nM T40954 CWO6S5 118366123 IC50 = 17.7 nM T40954 C3SW1L 122182611 IC50 > 100000 nM T40954 C6SUI3 122182612 IC50 > 100000 nM T40954 CSIV45 122182613 IC50 > 100000 nM T40954 CTW6P8 122182614 IC50 > 100000 nM T40954 CAL31C 122182615 IC50 > 100000 nM T40954 C9FKJ0 122182616 IC50 > 100000 nM T40954 CSKN75 122182617 IC50 = 820 nM T40954 C21KML 122182618 IC50 = 600 nM T40954 C5W2AZ 122182619 IC50 = 220 nM T40954 CCY8H4 122182620 IC50 = 320 nM T40954 CS4V9E 122182621 IC50 = 98 nM T40954 CZES29 122182622 IC50 = 250 nM T40954 CQ03EU 122182623 IC50 > 100000 nM T40954 CJ1O7X 122182624 IC50 > 100000 nM T40954 CM5B4S 122182625 IC50 > 100000 nM T40954 C12GHQ 122182626 IC50 > 100000 nM T40954 C10TBV 122182627 IC50 > 100000 nM T40954 C3PL6T 122182628 IC50 > 100000 nM T40954 C4U9MI 122184684 IC50 = 1700 nM T40954 CGR14F 127037772 IC50 = 20000 nM T40954 C7OWR2 127037773 IC50 = 20000 nM T40954 CWRH56 127038100 IC50 = 18000 nM T40954 C3OQ1G 127038116 IC50 = 20000 nM T40954 CBV1I2 127038367 IC50 = 20000 nM T40954 CLU2E5 127039056 IC50 = 15000 nM T40954 C2LXC6 127039373 IC50 = 20000 nM T40954 CO1DV3 127040391 IC50 = 10000 nM T40954 CNA9U5 127041463 IC50 = 20000 nM T40954 C37HMS 127041695 IC50 = 20000 nM T40954 CG47RT 130324335 IC50 = 6360 nM T40954 CV9PW4 130324347 IC50 = 3990 nM T40954 CMCO93 130324350 IC50 = 10800 nM T40954 CJZ2B5 130324358 IC50 = 31720 nM T40954 CIY63Q 130324359 IC50 = 6040 nM T40954 C9Z3XL 130324419 IC50 = 12120 nM T40954 C8C1OQ 130324429 IC50 = 9880 nM T40954 CYD48K 130324430 IC50 = 4810 nM T40954 CFJX81 130324435 Ki = 3430 nM T40954 C7H1ZA 130324436 IC50 = 13480 nM T40954 C7SO4Y 130324437 IC50 = 14910 nM T40954 C5NS9M 130324440 IC50 = 4980 nM T40954 CA4KB7 135411165 IC50 > 100000 nM T40954 C20SFP 135415592 IC50 = 407.38 nM T40954 C5U8SI 135416977 IC50 = 239.88 nM T40954 CPS4A8 135417221 Ki = 5700 nM T40954 CLZ2P8 135420365 IC50 = 15848.93 nM T40954 CU3KB8 135431348 IC50 = 1819.7 nM T40954 C27TMJ 135435089 IC50 = 30500 nM T40954 C7QOG3 135438127 Ki = 1860 nM T40954 CG7UC8 135439466 IC50 = 359 nM T40954 C2SL1G 135440025 Ki = 17700 nM T40954 CGN01S 135443857 IC50 = 310 nM T40954 C7GYM9 135449025 Ki = 176 nM T40954 C5ZXC3 135449835 IC50 = 25118.86 nM T40954 CJ68MB 135450778 Ki = 55.1 nM T40954 CZ8V4B 135457128 IC50 = 12589.25 nM T40954 C6AVP7 135461794 Ki = 490 nM T40954 C7NJF5 135462689 IC50 = 501.19 nM T40954 C3P9AV 135463610 IC50 > 100000 nM T40954 CWE78G 135463652 IC50 > 100000 nM T40954 CV3I9O 135463707 Ki = 77840 nM T40954 CN37YX 135464049 IC50 = 269.15 nM T40954 CB29QJ 135469329 Ki = 155 nM T40954 C0NR1W 135470528 IC50 = 1096.48 nM T40954 C90JVE 135471527 IC50 = 373 nM T40954 C7UG5Z 135473443 IC50 = 15848.93 nM T40954 COW48K 135479047 IC50 = 151.36 nM T40954 C7C8UR 135479918 IC50 = 1925 nM T40954 C68AMV 135480541 Ki = 25700 nM T40954 CPB61U 135480622 IC50 = 794.33 nM T40954 CC28JD 135491178 IC50 = 218.78 nM T40954 C5EO9Z 135492321 Ki = 890 nM T40954 CI8PN7 135513669 Ki = 160 nM T40954 CYPW68 135516658 Ki = 9.8 nM T40954 CFH2Z8 135529676 IC50 > 100000 nM T40954 C9PE7V 135581560 IC50 = 794.33 nM T40954 CJ1O3L 135590630 IC50 > 100000 nM T40954 CEA2Y4 135682068 IC50 > 100000 nM T40954 C62RLX 135724997 IC50 = 794.33 nM T40954 CGCX28 135773838 IC50 = 15848.93 nM T40954 CK6NE0 135973621 IC50 = 7943.28 nM T40954 CL49KZ 136026474 Ki = 4490 nM T40954 COAK95 136056475 IC50 = 1584.89 nM T40954 C92UKX 136087125 IC50 > 100000 nM T40954 CY36KX 136087126 IC50 > 100000 nM T40954 CYR3K4 136087127 IC50 > 100000 nM T40954 CWU02V 136097004 IC50 = 630.96 nM T40954 CXC4N5 136216653 IC50 = 20 nM T40954 CYNE32 136216654 IC50 = 140 nM T40954 CT8QA4 136216655 IC50 = 950 nM T40954 CW8L1R 136216656 IC50 = 1920 nM T40954 C20DTJ 136216657 IC50 = 6720 nM T40954 CSP97D 136216658 IC50 > 20000 nM T40954 CB08DP 136216659 IC50 = 2470 nM T40954 C71GCJ 136216660 IC50 = 16520 nM T40954 CW35IT 136216661 IC50 = 3650 nM T40954 C80HES 136216662 IC50 > 30000 nM T40954 CXQ69N 136216663 IC50 = 4950 nM T40954 C1C0AF 136216664 IC50 = 1630 nM T40954 CLI9P3 136216665 IC50 = 9240 nM T40954 C3KJ7C 136216666 IC50 = 2440 nM T40954 C41TAR 136216667 IC50 = 2100 nM T40954 C6YOF9 136216668 IC50 = 600 nM T40954 CY86RV 136223997 IC50 = 6.31 nM T40954 CN5A1G 136223998 IC50 = 6.31 nM T40954 CIMA43 136223999 IC50 = 794.33 nM T40954 C7M5YR 136224000 IC50 = 0.631 nM T40954 CS2CW1 136224230 IC50 = 1258.93 nM T40954 CWZ6T0 136224231 IC50 = 794.33 nM T40954 CEA92P 136224232 IC50 = 1.585 nM T40954 CG9B1W 136237996 IC50 = 1 nM T40954 CIF2G0 136240118 IC50 = 1.259 nM T40954 CBRF78 136241440 IC50 = 100 nM T40954 C8RVS3 136241441 IC50 = 1000 nM T40954 C0WRH3 136241442 IC50 = 501.19 nM T40954 CV7DF1 136241443 IC50 = 3.981 nM T40954 CW69SJ 136241444 IC50 > 100000 nM T40954 CQEF15 136241652 IC50 = 199.53 nM T40954 CZ5B8E 136245102 IC50 = 1.585 nM T40954 C6IYJ9 136245103 IC50 = 199.53 nM T40954 CAF69K 136245104 IC50 = 0.5012 nM T40954 CFP36E 136245105 IC50 = 501.19 nM T40954 CO04KE 136245106 IC50 = 1.259 nM T40954 CLC45W 136245107 IC50 = 19.95 nM T40954 CO0VQ2 136245108 IC50 = 501.19 nM T40954 C3Z0IY 136245109 IC50 = 794.33 nM T40954 C0D9ZF 136264296 IC50 = 10000 nM T40954 CV75NM 136326054 IC50 = 10960 nM T40954 CU5T0E 136326055 IC50 = 20890 nM T40954 CR9OM0 136599921 IC50 = 24260 nM T40954 CACM49 136748380 IC50 = 184 nM T40954 CFR34M 136859539 IC50 = 38 nM T40954 C9T7GL 136859540 IC50 = 32 nM T40954 C2OWB9 137631384 IC50 = 172 nM T40954 CC7OG9 137631566 IC50 = 385 nM T40954 CY7GA9 137632805 IC50 > 60000 nM T40954 C1W6UF 137632849 IC50 > 60000 nM T40954 CV47NQ 137633624 IC50 > 100000 nM T40954 CRM3Z7 137636550 IC50 = 7894 nM T40954 C3FP2H 137637320 IC50 > 60000 nM T40954 C2JB8X 137638109 IC50 > 60000 nM T40954 C7R8SO 137638384 IC50 = 37 nM T40954 C8N9JL 137638468 IC50 = 34 nM T40954 C7ORW6 137641987 IC50 = 117 nM T40954 C1U4SC 137642334 IC50 = 50240 nM T40954 C1NT8Q 137642531 IC50 = 60 nM T40954 C6WIM0 137642798 IC50 = 305 nM T40954 C5RH3O 137642939 IC50 = 247 nM T40954 C9ZT3C 137643234 IC50 = 5220 nM T40954 CK89RI 137644006 IC50 > 60000 nM T40954 CJ2ZB3 137645788 IC50 > 60000 nM T40954 CS79RN 137646442 IC50 = 61100 nM T40954 CWRC69 137646457 IC50 = 62 nM T40954 CG4NB3 137647236 IC50 > 60000 nM T40954 CP2AC4 137647881 IC50 = 4670 nM T40954 CFL54O 137648214 IC50 = 529 nM T40954 CMD09A 137648311 IC50 = 56680 nM T40954 C58OPE 137649016 IC50 = 55 nM T40954 C9A3JP 137650642 IC50 = 53 nM T40954 C4I9GC 137650872 IC50 = 103 nM T40954 C1BPK2 137651058 IC50 = 782 nM T40954 CBD2L3 137651750 IC50 = 223 nM T40954 CB15VR 137652637 IC50 = 41 nM T40954 C34ILA 137652722 IC50 = 86220 nM T40954 CD2IJ0 137653842 IC50 = 399 nM T40954 CKH7E6 137654238 IC50 > 60000 nM T40954 CN18YX 137655596 IC50 > 60000 nM T40954 C6T1WN 137655674 IC50 > 60000 nM T40954 C86KED 137656448 IC50 = 250 nM T40954 C8YD1I 137657260 IC50 = 41 nM T40954 CW20KA 137657391 IC50 = 33700 nM T40954 CC21KZ 137658196 IC50 = 70 nM T40954 CY7QC1 137658211 IC50 = 69 nM T40954 C97AUL 137658453 IC50 = 224 nM T40954 CWN5X3 137659818 IC50 > 60000 nM T40954 CX6O9I 137660389 IC50 = 77 nM T40954 CIE96G 137660639 IC50 > 60000 nM T40954 CSD2G0 137662251 IC50 = 57420 nM T40954 C2PU8Q 141538408 IC50 = 333 nM T40954 C1OS4B 141538409 IC50 = 322 nM T40954 C5N8QE 141538410 IC50 = 208 nM T40954 C3Q8PJ 141538411 IC50 = 292 nM T40954 CQ1AV7 141538412 IC50 = 510 nM T40954 CB0X8C 141538413 IC50 = 132 nM T40954 CNL1Y6 141538414 IC50 = 283 nM T40954 C94JGN 141538415 IC50 = 377 nM T40954 C2AQ8L 141538416 IC50 = 463 nM T40954 C8L9AO 141538417 IC50 = 138 nM T40954 CO5L3C 141538418 IC50 = 421 nM T40954 CUHI10 141538419 IC50 = 1130 nM T40954 CTDZ20 141538420 IC50 = 282 nM T40954 CHJW04 141538421 IC50 = 527 nM T40954 CPTC37 141538422 IC50 = 471 nM T40954 CQ5PJ2 141538425 IC50 = 674 nM T40954 C06GJX 141538426 IC50 = 417 nM T40954 CR19EQ 141538427 IC50 = 798 nM T40954 C0VBM8 145951102 IC50 = 95400 nM T40954 CA4M3S 145955768 IC50 = 27850 nM T40954 CTP64Q 145967497 Ki = 2890 nM T40954 C8F4OB 145967623 IC50 = 50500 nM T40954 C78CSF 145967638 IC50 = 25600 nM T40954 CB53JT 145967694 IC50 = 17500 nM T40954 CP1HE0 145968042 IC50 = 38800 nM T40954 C0NU8J 145968076 IC50 = 52500 nM T40954 C9SUO1 145968165 IC50 = 44300 nM T40954 CM7GB0 145968512 IC50 > 100000 nM T40954 CH2E4F 145968795 IC50 = 39100 nM T40954 CR1LX0 145969011 IC50 = 9800 nM T40954 C2YRN0 145969255 IC50 = 15200 nM T40954 CT30SC 145969792 IC50 = 48900 nM T40954 C0DG3T 145970254 IC50 > 100000 nM T40954 CN5VK7 145970362 IC50 > 100000 nM T40954 C6LIW3 145970385 IC50 = 20600 nM T40954 CZFI29 145970423 IC50 = 26900 nM T40954 CAQ9S1 145970624 IC50 > 100000 nM T40954 CF6YQ3 145970658 IC50 = 58100 nM T40954 C23CHM 145970797 IC50 = 11600 nM T40954 CC8T1Z 145987280 IC50 = 64300 nM T40954 CKBI34 145988409 IC50 = 17800 nM T40954 CRX3V8 145989045 IC50 = 15200 nM T40954 D00RIX 5280443 Ki = 520 nM T40954 D00YEV 5281605 IC50 = 2790 nM T40954 D01KKU 5281894 IC50 = 38000 nM T40954 D01UYI 5281607 IC50 = 840 nM T40954 D02JEZ 5281426 IC50 = 236000 nM T40954 D05WQF 637540 IC50 = 32.2 ug.mL-1 T40954 D06UEP 17027464 Ki > 30000 nM T40954 D07DJS 5280459 IC50 = 14740 nM T40954 D07YDN 5281654 IC50 = 2510 nM T40954 D09ALJ 5280805 IC50 = 52200 nM T40954 D09FDZ 5466139 IC50 = 6600 nM T40954 D0B5GC 11349 IC50 > 100000 nM T40954 D0D9OC 4584789 IC50 = 10190 nM T40954 D0E0RW 69894 IC50 = 138000 nM T40954 D0F1AS 80220 IC50 > 200000 nM T40954 D0G3TK 5280863 IC50 = 1060 nM T40954 D0IB3K 5320686 IC50 > 100000 nM T40954 D0J5DN 5284648 IC50 = 16800 nM T40954 D0MF5Y 5281614 IC50 = 4330 nM T40954 D0NJ4H 5281670 IC50 = 10100 nM T40954 D0PJ3M 637511 IC50 = 7.8 ug.mL-1 T40954 D0SY2M 5281708 IC50 = 429800 nM T40954 D0T2QL 444539 IC50 = 26.4 ug.mL-1 T40954 D0T3NP 7456 IC50 > 50000 nM T40954 D0T3PW 5281672 IC50 = 2380 nM T40954 D0V7AA 9064 IC50 > 100000 nM T40954 D0Y7HG 5281616 IC50 = 1800 nM T40954 D0YZ5G 5281416 IC50 = 8200 nM T40954 D0ZO1R 159460 IC50 > 100000 nM T10191 CR65YH 16134403 IC50 = 130 nM T10191 C39MQA 16134407 IC50 = 130 nM T10191 C15MYL 76311380 EC50 = 120000 nM T10191 C8OQV6 76311397 EC50 > 95000 nM T10191 C68XTR 76311401 EC50 > 37000 nM T10191 CB0AP7 76315000 EC50 = 73000 nM T10191 C3MP2V 76315002 EC50 > 29000 nM T10191 CQ8VB6 76315003 EC50 = 70400 nM T10191 CB6R4T 76318655 EC50 > 125000 nM T10191 C4TYD3 76322249 EC50 > 125000 nM T10191 CCO8S4 76322266 EC50 > 125000 nM T10191 C3RYP9 76325890 EC50 = 19900 nM T10191 C72JKF 76325893 EC50 = 122000 nM T10191 CONP50 76325897 EC50 = 22000 nM T10191 CCZ93B 76325920 EC50 > 66000 nM T10191 C40QTZ 76325926 EC50 > 100000 nM T10191 CXQ61N 76329481 EC50 > 62000 nM T10191 C4DS0Z 76329500 EC50 = 69600 nM T10191 CG45CZ 76333121 EC50 = 83800 nM T10191 CBQ02V 76336736 EC50 > 125000 nM T10191 CW12KH 76336764 EC50 = 4000 nM T10191 CE4R1M 90663470 IC50 = 130 nM T94444 D01XBA 5035 Ki = 0.87 nM T94444 D01ZII 2726 IC50 = 570 nM T94444 D02DPA 2756 Ki = 155000 nM T94444 D02HED 4748 IC50 = 33 nM T94444 D03GET 4055 IC50 = 200 nM T94444 D06NXY 5991 Ki = 430 nM T94444 D08QMX 5757 IC50 = 80 nM T94444 D09DWL 5719 Ki = 83000 nM T94444 D0AV3G 3151 Ki = 1200 nM T94444 D0E9CD 12127 IC50 = 15000 nM T94444 D0G9YH 2179 IC50 = 3200 nM T94444 D0Y2NE 448537 IC50 = 460 nM T94444 D0Z1RV 135398737 Ki = 5100 nM T94444 D0L4FS 5280961 IC50 = 340 nM T94444 C68LOU 1050 Ki = 30000 nM T94444 C5IOL8 4910 IC50 > 200000 nM T94444 C4DZ7E 82071 Ki = 1500000 nM T94444 CURQ71 151185 Ki = 100000 nM T94444 CZ9MO8 328856 Ki = 200000 nM T94444 CH9U5I 342159 Ki = 300000 nM T94444 CRE92U 358125 IC50 = 40 nM T94444 C5WFL2 11816380 Ki = 200000 nM T94444 C0GF4O 44333530 Ki = 300000 nM T94444 C9X2VD 44333855 Ki = 400000 nM T94444 D0O2DQ 237 IC50 = 3300 nM T11317 D0E6XR 3062316 Ki < 10 nM T11317 D0E3TC 44259 IC50 = 1.34 nM T11317 D0IQ0Z 46885626 IC50 = 70 nM T11317 CN8WB9 44189332 IC50 = 211 nM T11317 CV63UL 67240318 IC50 > 10000 nM T11317 C2MD1Q 155513187 IC50 > 10000 nM T11317 D0E7VO 59627005 IC50 = 5.5 nM T11317 D0US9O 45275255 IC50 = 190 nM T86264 C0XFA4 118725730 EC50 = 4.2 nM T86264 CZC20G 118725731 EC50 = 6.3 nM T86264 CAZ1C2 118725732 EC50 = 10.4 nM T86264 CGV5C6 118725733 EC50 = 12.6 nM T86264 C2G6IS 118725734 EC50 = 218.1 nM T86264 CA6VQ0 118725735 EC50 = 34 nM T86264 CCPA21 118725736 EC50 = 10 nM T86264 CQW8E3 118725737 EC50 = 8.4 nM T86264 CXNV46 118725738 EC50 = 1.1 nM T86264 C7G6SP 122191114 EC50 = 103.8 nM T86264 C7Q0XF 122191115 EC50 = 112.7 nM T86264 C9THL2 122191116 EC50 = 335.3 nM T86264 CX3C8Z 122191117 EC50 = 268.8 nM T86264 C0YL6N 122191118 EC50 = 164.5 nM T86264 CEH7I9 122191119 EC50 = 92.3 nM T86264 CDHS04 122191120 EC50 > 600 nM T86264 CZL7H2 122191121 EC50 = 369 nM T86264 CZ36PG 122191122 EC50 = 52.3 nM T86264 C0EM7S 122191123 EC50 > 600 nM T86264 CZBW79 122191124 EC50 = 458.3 nM T86264 CHDS85 122191127 EC50 = 300 nM T86264 CK06BZ 122192229 EC50 = 4.2 nM T86264 CAP8K5 122192230 EC50 > 600 nM T86264 CTY75A 122192231 EC50 > 600 nM T86264 C58QKF 122192232 EC50 > 600 nM T86264 CK6Y9H 122192233 EC50 = 585.6 nM T86264 C73WAT 122192234 EC50 = 272.2 nM T86264 C8WAO1 122192235 EC50 = 598.9 nM T86264 CKH7N5 122192236 EC50 > 600 nM T86264 C5CJR9 122192237 EC50 > 600 nM T86264 CM7EI4 122192238 EC50 = 477.4 nM T86264 CPAT35 122192239 EC50 = 516.9 nM T86264 C69OPR 122192240 EC50 > 600 nM T86264 CEZC35 122192242 EC50 = 531.7 nM T86264 C9BS3E 122192243 EC50 = 54.3 nM T86264 CU6RG2 122192244 EC50 = 75.1 nM T86264 C9YVD1 122192245 EC50 = 44.2 nM T86264 C1ZS6N 155525033 EC50 = 22 nM T86264 CEUH06 155543884 EC50 > 600 nM T86264 CV5MN6 155544304 EC50 = 21 nM T86264 CU8M5L 155554132 IC50 = 76 nM T86264 CID3L8 155554215 EC50 = 347 nM T55689 D0A8UP 10453818 IC50 = 1 nM T55689 CN3KA4 2743222 IC50 = 20 nM T55689 C1DPL5 2773253 IC50 = 130 nM T55689 C8SW7P 9808221 IC50 = 120 nM T55689 CSK87O 9813746 IC50 = 50 nM T55689 CBU19K 9814762 IC50 = 360 nM T55689 CFOX59 9818390 IC50 = 32 nM T55689 CG6W8R 9839754 IC50 = 1100 nM T55689 CQ3ED7 9856441 IC50 = 184 nM T55689 CD52YN 9878507 IC50 = 205 nM T55689 CG3CM8 9922280 IC50 = 6400 nM T55689 CMW0T9 9966186 IC50 = 19 nM T55689 C8FSI9 9968739 IC50 = 97 nM T55689 CH0R1M 10038557 IC50 = 3 nM T55689 CEKX28 10094001 IC50 = 170 nM T55689 CI70JE 10109540 IC50 = 23 nM T55689 CSX92P 10126521 IC50 = 1230 nM T55689 C1B9MQ 10150601 IC50 = 46 nM T55689 CA5J4V 10150622 IC50 = 8500 nM T55689 C36DNM 10215997 IC50 = 630 nM T55689 CCN87G 10267853 IC50 = 35 nM T55689 C27DUO 10268239 IC50 = 9952 nM T55689 CB2K1F 10287897 IC50 = 350 nM T55689 C41SEL 10293330 IC50 = 3 nM T55689 CV5B1A 10308583 IC50 > 5000 nM T55689 CJ0VN5 10310052 IC50 = 1500 nM T55689 CU21VN 10476544 IC50 = 250 nM T55689 CQ6V3T 10483172 IC50 = 200 nM T55689 CIP41D 11150497 IC50 = 900 nM T55689 C4EU7X 11188905 IC50 = 400 nM T55689 C9EMG6 11209350 IC50 = 4000 nM T55689 CZPB69 11210161 IC50 = 100000 nM T55689 CT4Y0D 11210560 IC50 = 160 nM T55689 C4N9ZL 11221206 IC50 = 100 nM T55689 C93CQK 11221441 IC50 = 100 nM T55689 CX6CF4 11232205 IC50 = 2000 nM T55689 CT38EP 11235216 IC50 > 50000 nM T55689 C5FO1B 11243200 IC50 > 50000 nM T55689 C6GHQ3 11244670 IC50 = 2000 nM T55689 CP6FX1 11268904 IC50 = 200 nM T55689 C2NRQ0 11270327 IC50 = 400 nM T55689 CAP59Z 11278342 IC50 = 210 nM T55689 C1JKX2 11290299 IC50 = 60 nM T55689 CXV91C 11304331 IC50 > 50000 nM T55689 CBL8D9 11314048 IC50 = 9000 nM T55689 CO5W9Q 11327297 IC50 = 700 nM T55689 CNTY27 11336871 IC50 = 600 nM T55689 CG91BA 11350292 IC50 = 9000 nM T55689 CAR45P 11359651 IC50 = 100 nM T55689 CL9G3Y 11425872 IC50 = 30 nM T55689 CF9M4R 11451482 IC50 = 300 nM T55689 CF4N7E 11486370 IC50 = 62 nM T55689 C7OPQ0 11772375 IC50 > 50000 nM T55689 C1R4MF 12995052 IC50 = 1500 nM T55689 C3Z4BI 22946387 IC50 = 52 nM T55689 C9F2ZH 22946388 IC50 = 15 nM T55689 C15ASX 23635398 IC50 > 50000 nM T55689 C9F1MQ 23635399 IC50 = 46 nM T55689 CXIA45 23635400 IC50 > 5000 nM T55689 CQ0H4M 23635401 IC50 > 5000 nM T55689 CZ5R6B 23635511 IC50 = 3200 nM T55689 C5S2QB 23635512 IC50 = 250 nM T55689 C4B8MX 23635513 IC50 = 680 nM T55689 CWD7J8 23635514 IC50 = 1100 nM T55689 C0ASM1 23635515 IC50 = 39 nM T55689 CKP70J 23635516 IC50 = 320 nM T55689 CM0X3T 23635632 IC50 = 26 nM T55689 C0VL9W 23635633 IC50 = 23 nM T55689 CJ73KM 23635634 IC50 = 2400 nM T55689 CWI26H 23635635 IC50 = 120 nM T55689 CP6J2G 23635636 IC50 = 210 nM T55689 C4GA2J 23635637 IC50 = 270 nM T55689 CT46CR 23635766 IC50 = 350 nM T55689 CVJ6C0 23635767 IC50 = 3100 nM T55689 CU61DC 23635768 IC50 = 3900 nM T55689 CF91IH 23635891 IC50 > 5000 nM T55689 CT67MK 23635892 IC50 = 1400 nM T55689 CKM0C8 23635893 IC50 = 23 nM T55689 CC1PX4 23635894 IC50 > 5000 nM T55689 C0XQ8E 23635895 IC50 = 65 nM T55689 CCPS26 23635896 IC50 > 5000 nM T55689 C4UY7R 23636019 IC50 = 250 nM T55689 CHTN58 23636020 IC50 = 71 nM T55689 CPV52Y 23636021 IC50 = 51 nM T55689 CD71KA 23636022 IC50 > 5000 nM T55689 C6QA3I 23636023 IC50 = 1100 nM T55689 CQ4U9X 23636024 IC50 = 110 nM T55689 C03PIO 44269054 IC50 = 48000 nM T55689 C8FV9I 44269065 IC50 = 5500 nM T55689 C4O3NC 44269084 IC50 = 8500 nM T55689 C5OMC2 44269096 IC50 > 100000 nM T55689 CYD78C 44269110 IC50 = 67000 nM T55689 C3YP4O 44269116 IC50 = 760 nM T55689 C3TRW9 44269136 IC50 = 1300 nM T55689 CU6FZ1 44269139 IC50 = 210 nM T55689 CL6Q5C 44293573 IC50 = 138 nM T55689 CJ9X3W 44293587 IC50 = 716 nM T55689 C5ZW4H 44293589 IC50 = 24 nM T55689 C83LXM 44293632 IC50 = 515 nM T55689 CW1R3C 44293704 IC50 = 47 nM T55689 C80MPQ 44293705 IC50 = 3200 nM T55689 CODV40 44293914 IC50 = 5 nM T55689 C6V8RJ 44294061 IC50 = 10 nM T55689 C48SBO 44336947 IC50 = 3 nM T55689 CDXL04 44336950 IC50 = 102 nM T55689 CCO9P3 44336955 IC50 = 28 nM T55689 C58KAQ 44336957 IC50 = 3 nM T55689 CRA03G 44337010 IC50 = 13 nM T55689 C9V6IF 44337054 IC50 = 18 nM T55689 C5GXI8 44337102 IC50 = 180 nM T55689 CT1BX8 44337103 IC50 > 1000 nM T55689 CM46SZ 44337107 IC50 = 7 nM T55689 CF9MH6 44337118 IC50 = 135 nM T55689 CM3IW2 44337143 IC50 = 75 nM T55689 CCX71W 44337144 IC50 = 5 nM T55689 CTE8Y2 44337145 IC50 = 20 nM T55689 C3B4LP 44337147 IC50 = 6 nM T55689 CNPW18 44337148 IC50 = 1270 nM T55689 C76TXC 44337149 IC50 = 6 nM T55689 CA6IN3 44337150 IC50 = 90 nM T55689 C1L0SI 44337151 IC50 = 6 nM T55689 C0B9HC 44337152 IC50 = 1 nM T55689 C1TZ7H 44337166 IC50 = 4 nM T55689 CW71UE 44337167 IC50 = 5 nM T55689 C4PAX6 44337168 IC50 = 111 nM T55689 C4RLD7 44337169 IC50 = 73 nM T55689 CO60HD 44337170 IC50 > 1000 nM T55689 CU35QX 44337194 IC50 = 1400 nM T55689 CF98ZA 44337197 IC50 = 4 nM T55689 C7O5NZ 44337204 IC50 > 1000 nM T55689 CG5MB4 44337206 IC50 = 7 nM T55689 CMKN89 44337210 IC50 = 14 nM T55689 C2FWP0 44337213 IC50 = 17 nM T55689 C0GV4I 44337214 IC50 = 240 nM T55689 CZ78GP 44337219 IC50 > 1000 nM T55689 C01CAD 44337220 IC50 = 98 nM T55689 C2D4MZ 44337221 IC50 = 55 nM T55689 CS5P0D 44337222 IC50 = 6 nM T55689 CBR16D 44337224 IC50 = 11 nM T55689 CG8T4S 44337225 IC50 = 8 nM T55689 CAEL40 44337226 IC50 = 5 nM T55689 C15OWY 44337238 IC50 = 10 nM T55689 CFGM76 44337241 IC50 = 0.2 nM T55689 C0K4YP 44337242 IC50 = 4 nM T55689 CE31HP 44337244 IC50 = 200 nM T55689 CWUV64 44337245 IC50 = 33 nM T55689 C7NFW3 44337256 IC50 = 2 nM T55689 CYC1R5 44337257 IC50 = 12 nM T55689 CX5M0T 44337279 IC50 > 1000 nM T55689 CCR01H 44337283 IC50 = 72 nM T55689 C4ENB5 44337294 IC50 = 120 nM T55689 CO07WF 44337298 IC50 = 9 nM T55689 CI7WN5 44337299 IC50 = 6 nM T55689 CQ4E6H 44337300 IC50 = 166 nM T55689 CDEY65 44337301 IC50 = 150 nM T55689 CLQ1T6 44337306 IC50 = 5 nM T55689 CU7PC0 44337307 IC50 = 250 nM T55689 CB9TJ6 44337309 IC50 = 17 nM T55689 CRVG32 44337310 IC50 = 60 nM T55689 CUJS96 44337317 IC50 = 150 nM T55689 CFO93X 44337318 IC50 > 1000 nM T55689 CF9UY8 44337323 IC50 > 1000 nM T55689 C8Q9PD 44337325 IC50 = 408 nM T55689 C5JE9A 44337329 IC50 = 4 nM T55689 C73JQF 44337331 IC50 = 160 nM T55689 CILP13 44337332 IC50 = 480 nM T55689 CZ8VQ7 44337335 IC50 = 180 nM T55689 C6W2BQ 44337339 IC50 = 2 nM T55689 CB5LF7 44337345 IC50 > 1000 nM T55689 C64NSB 44337346 IC50 = 246 nM T55689 C9GLD0 44337363 IC50 = 460 nM T55689 CQC5U6 44337364 IC50 = 7 nM T55689 CBZ3M6 44337365 IC50 = 326 nM T55689 C6ZK3U 44337376 IC50 > 1000 nM T55689 C08YMZ 44337377 IC50 > 1000 nM T55689 C10WEO 44337385 IC50 > 1000 nM T55689 CEG0Z6 44337422 IC50 = 314 nM T55689 CB3IV5 44337433 IC50 = 56 nM T55689 CNEY90 44337434 IC50 = 27 nM T55689 C06QIK 44337435 IC50 = 30 nM T55689 C6GV7S 44337504 IC50 = 62 nM T55689 CYGA20 44337505 IC50 = 900 nM T55689 CTVK89 44337506 IC50 = 93 nM T55689 C9KX0L 44337507 IC50 = 187 nM T55689 C7WXD0 44337521 IC50 = 51 nM T55689 C3J7IX 44337543 IC50 = 1 nM T55689 CW9BH3 44337544 IC50 = 8 nM T55689 C0NHI2 44435121 IC50 > 5000 nM T55689 CX7FC5 127052444 IC50 = 7 nM T55689 CPE25G 132569641 IC50 = 91 nM T55689 CA9HT3 132569642 IC50 = 2 nM T55689 CJZ72T 132609412 IC50 = 68 nM T55689 C2WQ3J 137634449 IC50 = 8 nM T55689 CIM69B 137635824 IC50 = 860 nM T55689 C7L3QJ 137635980 IC50 = 46 nM T55689 CA8JC3 137636332 IC50 = 110 nM T55689 C70IRM 137639760 IC50 = 130 nM T55689 CE25PO 137639805 IC50 = 810 nM T55689 C8MSZ5 137641307 IC50 = 20 nM T55689 CXT1C6 137644051 IC50 = 40 nM T55689 CI4O7W 137645324 IC50 = 180 nM T55689 C3FW6O 137645441 IC50 = 920 nM T55689 CQZ54F 137645671 IC50 = 19 nM T55689 CJ0ZT6 137646352 IC50 = 13 nM T55689 CM57XB 137646963 IC50 = 24 nM T55689 CC29QB 137647186 IC50 = 24 nM T55689 C6T7OZ 137647225 IC50 = 280 nM T55689 CK3I4O 137648814 IC50 = 810 nM T55689 C1P6YH 137649233 IC50 = 380 nM T55689 CU9PX7 137650998 IC50 = 570 nM T55689 CIP67Y 137652988 IC50 = 59 nM T55689 CXW5N8 137654706 IC50 > 5000 nM T55689 C7I5ZP 137656064 IC50 = 14 nM T55689 C0NAH1 137656573 IC50 = 100 nM T55689 C26BLP 137658606 IC50 = 16 nM T55689 CXZ3R4 137658655 IC50 = 230 nM T55689 C8KC5L 137659858 IC50 = 8 nM T55689 CF2O9Q 137660292 IC50 = 21 nM T55689 C2JM8S 137661297 IC50 = 1900 nM T76198 D0C7AA 5282440 IC50 > 100000 nM T76198 D0E3BH 5362391 IC50 = 1700 nM T76198 D0WL5V 9867642 Ki = 2.95 nM T76198 D00HTY 5280363 IC50 > 0.001 nM T76198 D00IQH 11677589 Ki > 5000 nM T76198 D00MZK 9911469 Ki > 10000 nM T76198 D0D9LB 6449876 IC50 = 11 nM T76198 D0GC5H 123879 Ki = 0.58 nM T76198 D0I3TU 45268455 Ki = 3804 nM T76198 D0K1EG 11508736 IC50 > 10000 nM T76198 D0LI1C 44469321 IC50 > 30000 nM T76198 D0RL4X 45270144 IC50 = 62600 nM T76198 D0SP5V 49843471 IC50 > 25000 nM T76198 D0X7EG 11462174 IC50 > 100000 nM T76198 D09AVU 46202376 IC50 = 7000 nM T76198 D03QGL 54343 Ki = 63 nM T76198 D03ZVW 6918030 IC50 = 12 nM T76198 D06UCV 23669776 IC50 = 360 nM T76198 D07JSK 51550 Ki = 650 nM T76198 D0H5PG 131717 IC50 = 6 nM T76198 D0K0VH 9867949 IC50 = 96 nM T76198 D0X8QI 3086644 Ki = 21 nM T76198 CYFR68 5036 Ki = 53 nM T76198 CJQE97 5581 Ki = 162.18 nM T76198 CAZT67 1283333 IC50 < 10000 nM T76198 CLM8P6 2114670 Ki > 25000 nM T76198 CUE37L 3077003 IC50 = 84 nM T76198 CI86PB 3078923 Ki = 6.8 nM T76198 CJ29HP 3078925 Ki = 5.7 nM T76198 COC2U7 3078928 Ki = 32 nM T76198 CR9T5W 3078930 Ki = 11 nM T76198 CK16QC 5311234 IC50 = 510 nM T76198 CO7N1Z 5311239 EC50 = 30000 nM T76198 CST20A 5311396 Ki = 2.7 nM T76198 CVY03O 5747298 IC50 = 970 nM T76198 CMG0X2 6366700 IC50 = 80 nM T76198 CH28KC 6366701 IC50 = 20 nM T76198 CY4N6E 6436053 IC50 = 19 nM T76198 CZ15QS 6441607 EC50 = 24 nM T76198 CV75GZ 6537211 IC50 = 380 nM T76198 C5P6IT 9801735 IC50 = 70 nM T76198 CURH60 9801972 Ki = 47 nM T76198 CQA35F 9802748 Ki = 3000 nM T76198 CT6JR1 9806791 Ki = 19054.61 nM T76198 C6TA3N 9809136 Ki = 3000 nM T76198 CV24TI 9817292 Ki = 4600 nM T76198 CHUM01 9825028 Ki = 39.4 nM T76198 CYNX09 9825293 EC50 = 2100 nM T76198 C96RQU 9865257 IC50 = 1160 nM T76198 C52IVO 9866368 IC50 = 1.1 nM T76198 C8J1XO 9868012 Ki = 100 nM T76198 C1L6XP 9871887 Ki = 46.77 nM T76198 CKMW12 9874010 Ki = 2100 nM T76198 CF0HC5 9888589 IC50 > 10000 nM T76198 CFC8G4 9894720 Ki > 3000 nM T76198 CA5N0K 9895436 Ki = 1100 nM T76198 CQ0X9R 9909510 IC50 > 10000 nM T76198 CUF02C 9910826 Ki = 150 nM T76198 CGLY84 9917280 Ki = 60255.96 nM T76198 CGT56V 9930263 IC50 = 17 nM T76198 C9UL7C 9930816 IC50 = 190 nM T76198 CJH36W 9931330 IC50 = 530 nM T76198 CZ5Q3U 9933925 Ki = 3600 nM T76198 CICE70 9938626 Ki = 2800 nM T76198 CH7PD4 9938840 IC50 = 16.4 nM T76198 CWDT69 9939791 Ki = 1500 nM T76198 C3LX4J 9953978 Ki = 230 nM T76198 C6SGH7 9954562 Ki > 500 nM T76198 C4UK2Q 9955802 Ki > 3000 nM T76198 C8ORC5 9971633 IC50 > 100000 nM T76198 CGI40J 9973005 IC50 = 73000 nM T76198 C7YR8X 9978044 Ki = 15 nM T76198 CQ8G2K 9978202 IC50 = 3280 nM T76198 CFD7S4 9978920 Ki = 3.6 nM T76198 CZQ0O9 9979675 IC50 = 330 nM T76198 C8WG6X 9980414 Ki = 5.1 nM T76198 CRI0K3 9981035 Ki > 74000 nM T76198 CDM12O 9983481 IC50 = 1100 nM T76198 CKN18V 9984004 Ki = 10 nM T76198 CG3M7O 10001037 Ki = 9.6 nM T76198 CZUJ52 10001608 IC50 > 10000 nM T76198 C7P9MS 10002804 IC50 = 1100 nM T76198 CCD24K 10007859 IC50 = 2.512 nM T76198 CG6FS1 10016908 IC50 > 100000 nM T76198 C6FG9T 10018213 IC50 = 19700 nM T76198 C7QL0V 10018589 IC50 = 295000 nM T76198 CR9E7U 10023102 IC50 = 280 nM T76198 C49HXB 10023647 Ki = 17 nM T76198 CB8Z2N 10024132 IC50 = 1900 nM T76198 CH10QM 10024143 IC50 = 70 nM T76198 CZ71TC 10024547 Ki = 1800 nM T76198 CTZQ75 10024655 Ki = 12 nM T76198 CMPT81 10025456 IC50 = 380 nM T76198 C85MLO 10026771 Ki = 2.2 nM T76198 CX4Q5E 10026942 Ki = 30 nM T76198 CUO4P3 10028328 IC50 = 12 nM T76198 CHN98V 10028338 Ki = 995 nM T76198 CS7ZB4 10028935 Ki = 14 nM T76198 CMQ93O 10029290 Ki = 92 nM T76198 CAJH39 10047167 Ki = 64 nM T76198 CQ3GW6 10047541 IC50 > 10000 nM T76198 C5RY8E 10047807 Ki = 11 nM T76198 CH3W6U 10047870 IC50 = 1200 nM T76198 CF1U8M 10050297 IC50 = 66 nM T76198 C8NTW2 10050347 IC50 = 21000 nM T76198 CP57DG 10050461 Ki = 3.7 nM T76198 CDX49N 10051178 Ki = 17 nM T76198 CW8MU3 10051348 IC50 = 42 nM T76198 CJP10L 10051943 Ki = 177.83 nM T76198 C9YBV0 10052055 IC50 = 340 nM T76198 C09LFU 10052612 IC50 = 51 nM T76198 CZW7P4 10067523 IC50 = 11000 nM T76198 CRW9E7 10071103 Ki = 30 nM T76198 C69ZDC 10071192 IC50 = 70 nM T76198 CRC31H 10072780 IC50 = 270 nM T76198 CM89DR 10073359 Ki = 24.5 nM T76198 C2X1PE 10074062 Ki = 164 nM T76198 CV48SW 10074101 Ki = 3.8 nM T76198 C6B0RS 10074652 IC50 = 19 nM T76198 C2MIC0 10074653 IC50 = 36 nM T76198 C49PUO 10074701 Ki = 15 nM T76198 C9KP4Y 10075114 IC50 = 300 nM T76198 CP68RF 10075294 IC50 = 28 nM T76198 CMJ87L 10087973 IC50 = 23400 nM T76198 CH1PV0 10092137 Ki = 46 nM T76198 CAF1N0 10092922 IC50 = 40 nM T76198 C9NPF7 10093386 Ki = 15 nM T76198 CGX84B 10094735 Ki = 10 nM T76198 CNE21V 10095268 Ki = 15.85 nM T76198 CK9F3Y 10095579 Ki = 47 nM T76198 CGBH15 10095993 IC50 = 33 nM T76198 CQ43YM 10096033 IC50 = 50 nM T76198 CV4TL1 10096378 IC50 = 74 nM T76198 C7H1AI 10096697 IC50 = 52 nM T76198 C2PIL6 10097814 Ki = 18 nM T76198 C3C9NH 10112823 Ki = 273 nM T76198 CRU76B 10114504 Ki = 363 nM T76198 CEX2R1 10116114 Ki = 260 nM T76198 C73CXR 10116116 Ki > 10000 nM T76198 C6JV2O 10136631 Ki = 136 nM T76198 CQGA49 10136760 Ki = 46 nM T76198 C0LDH4 10158956 Ki = 674 nM T76198 CAS19H 10161062 Ki = 219 nM T76198 CCEZ82 10162132 Ki = 250 nM T76198 CZR4A6 10181442 Ki = 11.7 nM T76198 C14ZJF 10204113 Ki = 484 nM T76198 C8CXL1 10204462 Ki = 226 nM T76198 CF1NB3 10207799 Ki = 120 nM T76198 CB7XJ2 10216985 Ki = 2.51 nM T76198 CF9G2A 10225819 Ki = 6972 nM T76198 C63UYT 10225820 Ki = 3190 nM T76198 CHM5I2 10226143 Ki = 17 nM T76198 CW94KD 10228100 Ki > 10000 nM T76198 C4C7UR 10244703 IC50 = 27300 nM T76198 C7AP9S 10244704 IC50 = 53100 nM T76198 C1BQ5M 10249316 Ki = 15 nM T76198 CK7YO0 10250339 IC50 = 3000 nM T76198 C0ED9Y 10251023 IC50 > 10000 nM T76198 CT5XI0 10251282 IC50 = 30 nM T76198 CH82JE 10251338 Ki = 7.6 nM T76198 CHD67V 10251769 Ki = 63 nM T76198 C1Q6IE 10251833 IC50 = 1300 nM T76198 C96QSH 10251861 Ki = 2.7 nM T76198 CLA94T 10253895 Ki = 6.1 nM T76198 C3CU7G 10254161 IC50 = 55 nM T76198 CLMR13 10254162 IC50 = 42 nM T76198 CNZI93 10254733 IC50 = 94 nM T76198 C8YHK7 10254794 Ki = 23.1 nM T76198 C3SO9M 10255332 IC50 = 170 nM T76198 CGS2U4 10256828 IC50 = 61 nM T76198 CD04FL 10258317 IC50 = 28 nM T76198 CK4C3W 10276571 Ki = 513 nM T76198 C1VIS5 10276868 Ki = 583 nM T76198 C8J9EN 10277744 Ki > 10000 nM T76198 CL7YG3 10287121 Ki > 13000 nM T76198 CD5Z7B 10297505 Ki = 200 nM T76198 CXKR41 10297616 Ki = 27.5 nM T76198 CQJI35 10299717 IC50 > 10000 nM T76198 CR86MT 10319482 Ki = 18 nM T76198 CT7K8Z 10320386 IC50 = 1200 nM T76198 CLQ96Z 10320883 IC50 = 7500 nM T76198 C4GU7S 10322452 Ki = 27 nM T76198 C5SY8E 10340286 IC50 = 120 nM T76198 C1PCZ7 10341794 IC50 = 140 nM T76198 CH01LV 10342027 IC50 = 230 nM T76198 CM7E1S 10342667 Ki = 171.6 nM T76198 CKAU36 10343670 IC50 = 210 nM T76198 C03LXV 10344641 IC50 = 2390 nM T76198 CWT1K9 10344683 Ki = 6887 nM T76198 CM1VU7 10345671 Ki = 35.7 nM T76198 CQE7L9 10345903 IC50 = 210 nM T76198 C95HPE 10347272 IC50 = 200 nM T76198 C8QHR9 10349225 Ki = 354.81 nM T76198 CH0L6C 10359399 Ki = 600 nM T76198 CE39GY 10363348 Ki = 23 nM T76198 CQ2FR8 10364232 Ki = 3.9 nM T76198 CD10ZM 10364364 IC50 = 520 nM T76198 CCSB81 10364780 Ki = 44 nM T76198 CKR60E 10365109 IC50 = 40 nM T76198 CR2I0W 10365193 Ki = 1.8 nM T76198 CYA20R 10365194 Ki = 9.5 nM T76198 C0YDL7 10366462 Ki = 7.7 nM T76198 CV46MX 10367685 IC50 = 230 nM T76198 CWR7X9 10369102 IC50 = 13 nM T76198 CU3TQ6 10369249 Ki = 0.91 nM T76198 CWZ14V 10370098 IC50 = 49 nM T76198 CK23JW 10371334 IC50 = 58 nM T76198 CY2JV4 10380987 IC50 = 74500 nM T76198 CX53ZT 10384315 IC50 = 360 nM T76198 CJ1QE0 10385168 IC50 = 29000 nM T76198 CWS2C6 10386146 Ki = 4 nM T76198 CSE10W 10386455 IC50 = 1040 nM T76198 C51JIX 10389527 EC50 > 20000 nM T76198 C2O6DR 10402602 IC50 = 46200 nM T76198 CEB37O 10402603 IC50 = 14700 nM T76198 CB19MW 10402929 Ki = 900 nM T76198 COH5S6 10406932 Ki = 15.3 nM T76198 CWC6S5 10407599 Ki = 29000 nM T76198 C1L7SZ 10409168 Ki = 37 nM T76198 CHVI06 10409291 Ki = 1300 nM T76198 CQU0V4 10409839 IC50 = 4160 nM T76198 CE2U6I 10410551 Ki = 280 nM T76198 C2BEN5 10411480 IC50 = 81 nM T76198 CFWJ57 10412393 Ki = 33 nM T76198 CX0MO5 10414389 Ki = 186.21 nM T76198 CDJ16L 10424476 IC50 = 49300 nM T76198 CS68RN 10430550 IC50 = 170 nM T76198 C4C6YG 10430971 Ki = 46 nM T76198 CIUY63 10431100 Ki = 8.3 nM T76198 C84KJB 10431401 IC50 = 970 nM T76198 C74EUN 10431402 IC50 = 160 nM T76198 CRFZ84 10432190 Ki = 78.9 nM T76198 CGT5X1 10433093 Ki = 387 nM T76198 CQG62B 10434230 IC50 = 60 nM T76198 C4GDE3 10436457 IC50 = 33 nM T76198 CNQ6T9 10448061 IC50 = 12200 nM T76198 C8WKX9 10451585 IC50 = 6000 nM T76198 CNK98U 10453182 IC50 = 880 nM T76198 CP8BJ9 10454345 Ki = 3.2 nM T76198 CF23ET 10454526 IC50 = 300 nM T76198 CYB1L0 10455115 IC50 = 170 nM T76198 C1VY2H 10455224 Ki = 77 nM T76198 COI27G 10456019 Ki = 88 nM T76198 CMC50K 10456399 Ki = 60 nM T76198 CBU8S9 10456444 Ki = 53 nM T76198 C85KTH 10457484 IC50 = 230 nM T76198 CHW12E 10458032 Ki = 64.8 nM T76198 CO8K7G 10458078 Ki = 17 nM T76198 C0X3OS 10458951 IC50 = 12 nM T76198 CKIH16 10460371 IC50 = 120 nM T76198 CI58CV 10476586 Ki = 4700 nM T76198 C5BS7K 10477535 Ki = 190 nM T76198 CJ9ZR7 10478975 Ki = 25 nM T76198 CJCL19 10479578 IC50 = 260 nM T76198 C7RJ5Y 10479865 IC50 = 21 nM T76198 C7W3DA 10480363 Ki = 4.2 nM T76198 CC83QY 10480515 Ki = 17.9 nM T76198 CYN53B 10480645 Ki = 6.1 nM T76198 CJ2T5E 10483231 IC50 = 62 nM T76198 CZ1XW6 10483360 IC50 = 30000 nM T76198 CU90BJ 10494367 IC50 = 3000 nM T76198 CB42FY 10495597 Ki = 338.84 nM T76198 CA8CF2 10500543 IC50 = 21000 nM T76198 CYTV60 10502508 IC50 = 210 nM T76198 C39BYU 10502610 IC50 = 670 nM T76198 C60WMU 10503252 IC50 = 130 nM T76198 C68XED 10503638 IC50 = 300 nM T76198 C18NWE 10518243 IC50 = 71000 nM T76198 C3TY0D 10518244 IC50 = 30000 nM T76198 CUFL39 10524500 IC50 = 18 nM T76198 C9IU3F 10526115 IC50 = 330 nM T76198 C3XID0 10526677 IC50 = 47 nM T76198 CZ2H8E 10529261 IC50 = 240 nM T76198 C4F9MA 10529683 IC50 = 740 nM T76198 CBPQ89 10542153 IC50 = 13000 nM T76198 C54MEV 10543197 IC50 = 7100 nM T76198 CUC93I 10545734 IC50 = 35 nM T76198 C16GTM 10546960 IC50 = 61 nM T76198 CANM20 10547489 IC50 = 2100 nM T76198 CF4G6L 10548488 IC50 = 81 nM T76198 C01LER 10548754 Ki = 1000 nM T76198 CW73IA 10550018 IC50 = 27 nM T76198 CTY02L 10552450 IC50 = 150 nM T76198 C58ZOU 10552612 IC50 = 280 nM T76198 C2C1VJ 10552843 IC50 = 83 nM T76198 C9XUE2 10577317 Ki = 5370.32 nM T76198 C23AHC 10590325 Ki = 9549.93 nM T76198 CRU0P1 10591274 IC50 = 7700 nM T76198 CMO37F 10594576 IC50 = 3100 nM T76198 C3GKS1 10595288 IC50 = 810 nM T76198 CJ7IT3 10599289 IC50 = 410 nM T76198 CD1V5X 10601327 IC50 = 110 nM T76198 CMY4P3 10601359 IC50 > 10000 nM T76198 CQ0PC7 10619606 IC50 = 120 nM T76198 CZT9C2 10620837 IC50 = 38 nM T76198 CPV7D6 10623568 IC50 = 1100 nM T76198 CEC6Q0 10637870 IC50 = 33000 nM T76198 CH1VS3 10637871 IC50 = 20000 nM T76198 CD13GN 10648014 IC50 = 1300 nM T76198 CI5HA0 10648334 IC50 > 10000 nM T76198 CX1R3B 10661867 IC50 = 24000 nM T76198 CGRY48 10669025 IC50 = 11 nM T76198 C4NGP3 10669026 IC50 = 7 nM T76198 CUD90Y 10669649 IC50 = 30 nM T76198 CN05QE 10670440 IC50 = 77 nM T76198 C9YQG5 10670992 IC50 > 10000 nM T76198 C9SUW2 10671942 IC50 = 1700 nM T76198 COEL58 10683471 Ki = 34673.69 nM T76198 CYGK01 10686657 IC50 = 8800 nM T76198 CL8OZ7 10686658 IC50 = 5000 nM T76198 C3WRM7 10696132 IC50 = 1300 nM T76198 C0K1ZP 10697301 IC50 = 55 nM T76198 C7H8NA 10717385 IC50 = 0.13 nM T76198 CT14ZS 10717572 IC50 = 1300 nM T76198 C6DPF4 10717914 IC50 = 32 nM T76198 C7GY6X 10739351 IC50 > 10000 nM T76198 CY8IB2 10740699 IC50 > 10000 nM T76198 C12SBH 10741017 IC50 > 10000 nM T76198 CG17HE 10741197 IC50 > 10000 nM T76198 C1ICD7 10741449 IC50 = 830 nM T76198 CK8O4Z 10741899 IC50 = 430 nM T76198 CU2LS0 10742144 Ki = 16218.1 nM T76198 C3QZJ8 10756559 IC50 = 7200 nM T76198 C1PHY8 10756560 IC50 = 104000 nM T76198 C53NGA 10756561 IC50 = 47000 nM T76198 CM51CL 10761205 IC50 = 16 nM T76198 CMF5P7 10762387 IC50 = 1100 nM T76198 CTBF04 10762411 IC50 = 1300 nM T76198 CVQ3J9 10764618 IC50 = 1000 nM T76198 C3AJ5O 10764758 IC50 = 610 nM T76198 C17OLN 10766313 IC50 = 330 nM T76198 C64MLE 10767455 IC50 = 1200 nM T76198 C4AB0L 10780482 IC50 = 15000 nM T76198 CF5E4M 10786712 IC50 = 1700 nM T76198 C2MBK5 10789142 Ki = 1479.11 nM T76198 CD1YX8 10813802 IC50 = 270 nM T76198 C8CV6J 10827996 IC50 = 25000 nM T76198 CXZ15O 10833696 IC50 = 21000 nM T76198 C14SCL 10834286 Ki = 83176.38 nM T76198 CTOQ40 10852668 IC50 = 25000 nM T76198 CKST02 11122314 IC50 > 10000 nM T76198 C7H3LX 11166017 Ki = 2500 nM T76198 CRI92F 11189801 Ki = 12183 nM T76198 CF0M3A 11201307 Ki = 26 nM T76198 C61PSW 11201693 Ki > 15000 nM T76198 CU7NJ3 11202399 Ki = 51 nM T76198 C12OPV 11237257 Ki = 4.3 nM T76198 C4S5MX 11249458 Ki > 10000 nM T76198 CIH90K 11259797 Ki = 184 nM T76198 C0LNI5 11260506 Ki = 180 nM T76198 C6ZOS1 11261579 Ki = 4.5 nM T76198 C70ESM 11269563 Ki = 14 nM T76198 CW3IZ0 11270709 Ki = 520 nM T76198 C8Y5TV 11282319 Ki = 88 nM T76198 CQ2V3R 11282605 Ki > 15000 nM T76198 CJ2V7N 11292620 Ki = 5100 nM T76198 CZU2D7 11293771 Ki > 10000 nM T76198 C9E4SW 11294166 Ki = 7100 nM T76198 CBJ75S 11294992 Ki = 138 nM T76198 C60SAH 11316066 Ki = 310 nM T76198 C8D5JF 11318288 Ki = 150 nM T76198 C4GC1Y 11350967 Ki = 3100 nM T76198 CP8L6Q 11364260 Ki > 5900 nM T76198 C4LJ3B 11374485 Ki = 390 nM T76198 CTHZ75 11374965 Ki = 78 nM T76198 CJ90WI 11386109 Ki = 130 nM T76198 CN2TG7 11387144 Ki > 1000 nM T76198 CWHO39 11407826 Ki = 3100 nM T76198 CXPO04 11408533 Ki = 1200 nM T76198 C6QLE7 11452761 Ki > 20000 nM T76198 CUB3R5 11454655 Ki = 72 nM T76198 CZ4K0P 11476788 Ki = 168 nM T76198 CE2JA4 11488860 Ki = 338 nM T76198 CW3YO5 11494768 IC50 > 25000 nM T76198 CH6U3F 11502680 IC50 = 0.65 nM T76198 CQ6IU7 11509269 IC50 > 25000 nM T76198 C0HFN7 11510008 IC50 = 45.53 nM T76198 CS2LR0 11516353 IC50 > 25000 nM T76198 CSK1M2 11531590 IC50 = 0.7 nM T76198 CF2OM8 11539410 IC50 > 25000 nM T76198 C2B8HY 11545850 Ki = 540 nM T76198 CM7HK0 11551847 IC50 > 25000 nM T76198 CD15FQ 11567679 IC50 = 1.26 nM T76198 CU2FH8 11568248 IC50 = 1.48 nM T76198 C0IY9D 11568384 IC50 = 1.17 nM T76198 C1W2ZK 11577792 Ki > 6000 nM T76198 CM7S6Q 11588648 Ki > 10000 nM T76198 C7Y6XJ 11597294 Ki = 0.84 nM T76198 CE6G3Y 11604299 IC50 = 0.71 nM T76198 C2M8HZ 11610353 IC50 > 25000 nM T76198 C9L5VD 11631813 IC50 > 25000 nM T76198 CD7R5P 11631965 IC50 > 25000 nM T76198 CD9MI2 11633163 IC50 = 2530 nM T76198 C3GYL1 11633215 IC50 = 55.17 nM T76198 CV3D4O 11647396 IC50 = 38.52 nM T76198 CMB6F9 11653874 IC50 > 25000 nM T76198 CX9BC0 11656254 IC50 = 126.28 nM T76198 CO3XR6 11661725 IC50 = 0.56 nM T76198 C0YP8G 11662021 IC50 = 0.7 nM T76198 C51UDK 11667741 IC50 > 10000 nM T76198 CWDP63 11676121 IC50 = 2.65 nM T76198 C2YR5H 11676145 IC50 = 181 nM T76198 C72BNQ 11682521 IC50 > 25000 nM T76198 CS3DL1 11683470 IC50 = 0.79 nM T76198 CW8RY9 11689895 IC50 > 25000 nM T76198 C9CM2R 11695689 IC50 > 25000 nM T76198 C3BSV4 11696697 Ki > 13000 nM T76198 C85JBY 11697902 IC50 = 2.68 nM T76198 CY02HC 11704760 IC50 = 1.58 nM T76198 CCJ5S3 11723604 IC50 = 23900 nM T76198 CAB5I6 11741746 Ki = 2813 nM T76198 C5QS6Y 11742649 Ki = 646.4 nM T76198 CEJD82 11742673 Ki = 6 nM T76198 CNYK74 11743212 Ki = 400 nM T76198 C3OW1Z 11743676 Ki = 2081 nM T76198 CV0T6Z 11744062 Ki = 3.4 nM T76198 C2ELZ1 11744063 Ki = 6.1 nM T76198 C8E4PV 11750835 Ki = 3100 nM T76198 C5LMZ4 11753841 IC50 = 12 nM T76198 C9LXS2 11754856 IC50 = 3000 nM T76198 CM3B0K 11755215 IC50 = 26 nM T76198 CXW63P 11755659 IC50 = 25 nM T76198 CX3ZO1 11755897 Ki = 14 nM T76198 CRDO34 11756528 Ki = 20 nM T76198 CT34LO 13230981 Ki > 13000 nM T76198 CAMR49 13720716 IC50 = 39810.72 nM T76198 C7WS8H 13720717 IC50 = 2454.71 nM T76198 CO19GA 14372497 Ki = 1.7 nM T76198 C93KFC 14372503 Ki = 990 nM T76198 C69REM 14372504 Ki = 2.6 nM T76198 CC68GR 14372505 Ki = 172 nM T76198 CJK30Q 14953067 Ki = 23 nM T76198 CXP81B 14953071 Ki = 670 nM T76198 CIP5D0 14953072 Ki = 7.8 nM T76198 CM1YA0 14953073 Ki = 52 nM T76198 CA8V1M 14953075 Ki = 870 nM T76198 CVGS75 14953076 Ki = 5600 nM T76198 CH2E5Y 14953077 Ki = 1700 nM T76198 C5URS0 14953078 Ki = 31 nM T76198 CSNR71 14953080 Ki = 160 nM T76198 CH09GK 14953084 Ki = 23 nM T76198 C0U8VZ 14953086 Ki = 6 nM T76198 CZ8B1O 14953087 Ki = 5 nM T76198 C7MH5C 14953088 Ki = 15 nM T76198 CLIC40 14953089 Ki = 12 nM T76198 CK8U3G 14953090 Ki = 4 nM T76198 C5R2YM 14953092 Ki = 12 nM T76198 C3FL4N 14953093 Ki = 6 nM T76198 C7HO3T 14953096 Ki = 13 nM T76198 COB8P0 14953097 Ki = 20 nM T76198 C8UEO5 14953098 Ki = 37 nM T76198 C2EW7V 14953103 Ki = 31 nM T76198 CY18QP 14953104 Ki = 16 nM T76198 CEB32X 14953106 Ki = 60 nM T76198 CFL0C8 14953108 Ki = 11 nM T76198 CG46HN 14953114 Ki = 39 nM T76198 CSE3Q6 14953115 Ki = 7 nM T76198 C7QX8V 14953120 Ki = 140 nM T76198 CTAU25 15018450 IC50 = 260 nM T76198 CPY35L 15018454 IC50 = 1100 nM T76198 CF91SO 15018459 IC50 = 540 nM T76198 CEJB18 15018463 IC50 = 2400 nM T76198 C6ST0N 15125130 IC50 = 30 nM T76198 CW3HB6 15125138 IC50 = 4.4 nM T76198 CBD64J 15157534 Ki = 2.4 nM T76198 CHW6G0 15157538 Ki = 2.2 nM T76198 CB8ZE9 15157541 Ki = 9.1 nM T76198 CILK97 15291968 IC50 = 2.6 nM T76198 C06OGJ 15486805 IC50 = 6909 nM T76198 C0L3VU 15486806 IC50 > 10000 nM T76198 CWQ8B9 15551228 Ki > 500 nM T76198 C8SP6X 15680093 Ki = 42 nM T76198 C4ML2W 15745526 IC50 = 1700 nM T76198 CQ4SA3 15745527 IC50 = 100 nM T76198 CK6UH8 15749427 Ki > 1000 nM T76198 CIS83K 15947857 Ki = 39 nM T76198 C3L0RK 15948325 Ki = 630 nM T76198 CM7J9N 16049493 Ki = 130 nM T76198 CFN1T4 16219283 IC50 = 31 nM T76198 CRZT49 16222207 IC50 = 31000 nM T76198 CI61TE 16678098 IC50 > 10000 nM T76198 CR34WC 16755884 IC50 = 99 nM T76198 CPT40Q 16755885 IC50 = 528 nM T76198 CMQR02 16756877 IC50 = 8750 nM T76198 CNV6L7 16756977 IC50 = 233 nM T76198 C7JSW0 16756978 IC50 = 155 nM T76198 CBV1G3 16756979 IC50 = 843 nM T76198 CC10OK 16756980 IC50 = 151 nM T76198 CE6AH2 16756981 IC50 = 423 nM T76198 CC7LE1 16756982 IC50 = 413 nM T76198 C9C1YU 16757078 IC50 = 120 nM T76198 C5EUX8 16757079 IC50 = 387 nM T76198 CIO5F4 16757080 IC50 = 201 nM T76198 CFR59W 16757081 IC50 = 400 nM T76198 CYMU04 16757082 IC50 = 95 nM T76198 C8ZWJ9 16757083 IC50 = 401 nM T76198 CZSB30 16757174 IC50 = 152 nM T76198 CK17JG 16757175 IC50 = 446 nM T76198 CRM20S 16757176 IC50 = 4840 nM T76198 CEWO04 16757177 IC50 = 749 nM T76198 CA28CP 16757178 IC50 = 111 nM T76198 C1HVD4 16757179 IC50 = 565 nM T76198 C5K8ZC 16757268 IC50 = 2080 nM T76198 CUV74O 16757375 IC50 = 42 nM T76198 CIX13C 16757376 IC50 = 2640 nM T76198 C2X5QT 16757377 IC50 = 17 nM T76198 CI8X7C 16757378 IC50 = 4220 nM T76198 CX7LE5 16757379 IC50 = 59 nM T76198 C30YTQ 16757380 IC50 = 523 nM T76198 CQSG13 16757381 IC50 = 2420 nM T76198 C8S4UD 16757483 IC50 = 698 nM T76198 CJL24R 16757484 IC50 = 98 nM T76198 CHY18C 16757485 IC50 = 885 nM T76198 CZ8Y6E 16757486 IC50 = 302 nM T76198 C8FRJ6 16757487 IC50 = 875 nM T76198 C1X6JH 16757488 IC50 = 1100 nM T76198 CK69TB 18476686 Ki = 200 nM T76198 CTX30D 18944131 IC50 = 130 nM T76198 CE3F5N 19097508 IC50 = 7 nM T76198 CGF28X 21019821 Ki = 200 nM T76198 CX08BC 21198692 Ki > 500 nM T76198 CPMI48 22083972 Ki = 16000 nM T76198 CBW0P7 22083975 Ki = 2300 nM T76198 C4SVP2 22083978 Ki = 730 nM T76198 CL1GO3 22882094 IC50 = 190 nM T76198 C35UQD 22882095 IC50 = 600 nM T76198 CZE62L 22882098 IC50 = 600 nM T76198 CVQK41 22882109 IC50 = 20 nM T76198 CRJ29A 22882110 IC50 = 60 nM T76198 C1SW6Y 22901615 IC50 = 9 nM T76198 CT84KG 23276768 IC50 = 1800 nM T76198 C43IRD 23276769 IC50 = 52000 nM T76198 C7CS3T 23276770 IC50 = 2500 nM T76198 CJ5CI8 23276771 IC50 = 1500 nM T76198 CF81SW 23582412 IC50 > 10000 nM T76198 CP2S4J 23663736 Ki = 930 nM T76198 C3BLZ2 23673317 IC50 = 950 nM T76198 CYB19L 23679440 IC50 = 1340 nM T76198 C9H4WT 23686961 Ki = 316.23 nM T76198 CASU54 23696973 Ki = 10 nM T76198 CKWG61 23705162 Ki = 15 nM T76198 C8X0BG 23964891 Ki = 6100 nM T76198 C42LYP 24765153 Ki = 5039 nM T76198 CF72YI 24765671 Ki >= 785 nM T76198 C31JZP 24765672 Ki >= 2500 nM T76198 C4QX7Y 24765675 Ki >= 930 nM T76198 CL7Z9U 24765768 Ki >= 110 nM T76198 CFQA40 24952577 Ki > 7282 nM T76198 CD98IN 24952580 Ki > 456 nM T76198 C81WVN 24952927 Ki > 5474 nM T76198 CZT83E 24952928 Ki > 501 nM T76198 C8YHX3 24953283 Ki > 224 nM T76198 CZ93FO 24953285 Ki > 628 nM T76198 C17JTY 24953286 Ki > 2226 nM T76198 CFT0W5 24953624 Ki > 4992 nM T76198 C42VMD 24953625 Ki > 3461 nM T76198 C7B2EW 24953628 Ki > 2117 nM T76198 CXQJ67 25002382 Ki >= 1291 nM T76198 CN5SH9 25003075 Ki = 6700 nM T76198 CEX34J 25817650 Ki = 6852 nM T76198 CI90SE 35028115 Ki = 1050 nM T76198 C8R2PE 40517075 Ki = 4200 nM T76198 CNOF71 44138108 Ki = 935 nM T76198 C5G4LN 44159411 IC50 = 67400 nM T76198 CHI65U 44159530 IC50 = 23000 nM T76198 CMNH53 44159772 IC50 = 11300 nM T76198 C2AV1K 44190762 IC50 = 2030 nM T76198 CZ29JY 44205724 IC50 = 63700 nM T76198 CYH56D 44210947 IC50 = 330 nM T76198 CR68BA 44250281 Ki > 10000 nM T76198 CN90FE 44269464 Ki > 13000 nM T76198 C1L0ET 44269468 Ki > 13000 nM T76198 C5KRQ4 44269486 Ki > 13000 nM T76198 CL6M2P 44269516 Ki > 13000 nM T76198 CON8R9 44269520 Ki > 13000 nM T76198 C6MBG0 44269521 Ki > 13000 nM T76198 CZ3Q1L 44269523 Ki > 13000 nM T76198 CRL61O 44269532 Ki > 13000 nM T76198 C1Z4LU 44269540 Ki > 13000 nM T76198 CM72FA 44269542 Ki > 13000 nM T76198 CN0JV2 44269543 Ki > 13000 nM T76198 C28UJH 44269544 Ki > 13000 nM T76198 CR1IY6 44269568 Ki > 13000 nM T76198 CI3C9O 44269596 Ki > 13000 nM T76198 CC0EW9 44269597 Ki > 13000 nM T76198 CD7AP4 44271646 Ki = 810 nM T76198 CY67ID 44271957 Ki = 510 nM T76198 C5XR1B 44273260 IC50 = 6000 nM T76198 CD59EH 44273351 IC50 = 1800 nM T76198 CH5TE2 44273387 IC50 = 1900 nM T76198 C3M8UJ 44273402 IC50 = 650 nM T76198 C5ZD9O 44273404 IC50 = 1900 nM T76198 C89MWE 44273412 IC50 = 650 nM T76198 C48QMN 44273414 IC50 = 1800 nM T76198 C0AW8H 44273415 IC50 = 1800 nM T76198 CRX3B2 44273434 IC50 = 200 nM T76198 CJ9Q6N 44273435 IC50 = 1700 nM T76198 C9C1UF 44273436 IC50 = 5500 nM T76198 C9P1SF 44273447 IC50 = 630 nM T76198 CXGH71 44273448 IC50 = 1800 nM T76198 CU5C6G 44273449 IC50 = 1800 nM T76198 CKYM27 44273462 IC50 = 2200 nM T76198 CYEZ79 44273463 IC50 = 4700 nM T76198 C1D3RQ 44273464 IC50 = 2000 nM T76198 CT5WB9 44273474 IC50 = 1900 nM T76198 C5T3EF 44273475 IC50 = 650 nM T76198 C2QR6B 44273483 IC50 = 680 nM T76198 CM07GJ 44273488 IC50 = 4400 nM T76198 CR8L6Q 44273489 IC50 = 250 nM T76198 CYD9Z1 44273497 IC50 = 210 nM T76198 C9FBU2 44273498 IC50 = 560 nM T76198 CI3FW2 44273499 IC50 = 1600 nM T76198 C6CTM3 44273500 IC50 = 750 nM T76198 CHF1B2 44273502 IC50 = 1900 nM T76198 CN4WL8 44273506 IC50 = 2300 nM T76198 CXP20B 44273521 IC50 = 1800 nM T76198 C2GPE0 44273522 IC50 = 1900 nM T76198 C1XWJ8 44273523 IC50 = 1900 nM T76198 C8LG0Z 44273524 IC50 = 600 nM T76198 CLB4X5 44273538 IC50 = 620 nM T76198 C9Z7CW 44273539 IC50 = 600 nM T76198 CV42TJ 44273540 IC50 = 200 nM T76198 CEU7G0 44273541 IC50 = 20000 nM T76198 CKA4W3 44273542 IC50 = 1700 nM T76198 C7IJ8D 44273570 IC50 = 1800 nM T76198 CB6I5R 44273574 IC50 = 2000 nM T76198 CRQJ86 44273588 IC50 = 1900 nM T76198 C75AWE 44273591 IC50 = 1300 nM T76198 CUA86I 44273742 IC50 = 1700 nM T76198 C9E4GN 44273778 IC50 = 2000 nM T76198 CTY40V 44273780 IC50 = 1900 nM T76198 C3D8MA 44273792 IC50 = 200 nM T76198 CTO91G 44273796 IC50 = 2000 nM T76198 C5QLK6 44273805 IC50 = 2000 nM T76198 CWJC89 44285146 IC50 > 10000 nM T76198 C5P9CF 44285208 IC50 > 10000 nM T76198 CCD2S1 44285209 IC50 > 10000 nM T76198 C9U7YH 44285251 IC50 > 10000 nM T76198 C6EZ1R 44285252 IC50 > 10000 nM T76198 CS64GQ 44285310 EC50 > 20000 nM T76198 CDP9F2 44285328 IC50 > 10000 nM T76198 CR12GY 44293931 IC50 = 1980 nM T76198 CLQ5W7 44304222 IC50 = 6000 nM T76198 C7BOQ6 44304226 IC50 = 6500 nM T76198 CIN1L5 44304262 IC50 = 1400 nM T76198 CX2P8G 44304264 IC50 = 180 nM T76198 C89CAK 44304265 IC50 = 1700 nM T76198 CM7V1R 44304271 IC50 = 180 nM T76198 C2C5LN 44304296 IC50 = 5200 nM T76198 CES76C 44304297 IC50 = 1800 nM T76198 COSQ63 44304350 IC50 = 12000 nM T76198 CF9T3N 44304384 IC50 = 130 nM T76198 CRE2V1 44304473 IC50 = 2300 nM T76198 CYDH52 44304559 IC50 = 60 nM T76198 C46GHR 44304640 IC50 = 9000 nM T76198 CS4JV9 44304641 IC50 = 200 nM T76198 C3ACZ5 44304642 IC50 = 1600 nM T76198 C40FNQ 44304706 IC50 = 26000 nM T76198 CZ4GJ7 44305326 IC50 = 46 nM T76198 CS0YH6 44305343 IC50 = 22 nM T76198 C9O7JM 44305452 IC50 = 228 nM T76198 C4GLA1 44305478 IC50 = 24 nM T76198 C92WKH 44305481 IC50 = 57 nM T76198 CFQ9O3 44305522 IC50 = 510 nM T76198 CG2OL4 44305538 IC50 = 88 nM T76198 CB62ZJ 44305550 IC50 = 795 nM T76198 CT2CF5 44305675 IC50 = 18 nM T76198 CWZJ12 44305824 IC50 = 820 nM T76198 CV9WB4 44306573 EC50 = 24 nM T76198 CB6SA5 44306604 EC50 = 3110 nM T76198 C8WIK3 44310390 IC50 = 20 nM T76198 CX1AW6 44310394 IC50 = 200 nM T76198 C8P9YM 44331597 Ki = 625 nM T76198 C91KOE 44333604 IC50 = 25000 nM T76198 C9ZH7J 44338130 Ki > 73000 nM T76198 CH2VD3 44338186 Ki > 73000 nM T76198 CXPZ62 44338224 Ki > 70000 nM T76198 CPW0H6 44338236 Ki = 2000 nM T76198 CXEQ14 44338237 Ki = 2000 nM T76198 C92LYP 44338257 Ki = 950 nM T76198 C7CKX5 44338263 Ki = 1500 nM T76198 CQHD85 44338264 Ki > 74000 nM T76198 CW8A4D 44338272 Ki = 1500 nM T76198 CYP6X3 44338285 Ki = 3800 nM T76198 C8R3HT 44338286 Ki = 11900 nM T76198 CX5Y0E 44338291 Ki = 3100 nM T76198 CW0EV9 44338292 Ki = 7000 nM T76198 CWM3S8 44338297 Ki = 4000 nM T76198 CGET31 44338308 Ki = 900 nM T76198 CVZM05 44338310 Ki > 75000 nM T76198 C85MCE 44338319 Ki = 6000 nM T76198 CC1D4E 44338326 Ki = 2200 nM T76198 CV37EY 44338387 Ki = 9100 nM T76198 C2ODN5 44338389 Ki = 9300 nM T76198 CWYD83 44338402 Ki > 71000 nM T76198 CCG6V3 44344457 IC50 = 44 nM T76198 C7VZ2Y 44346027 IC50 > 100000 nM T76198 CW8XQ9 44350662 IC50 = 100 nM T76198 CYCS78 44350670 IC50 = 130 nM T76198 CEVM75 44353026 IC50 = 6600 nM T76198 C8FWC9 44353027 IC50 = 100000 nM T76198 CQ5S9G 44353042 IC50 = 360 nM T76198 CWP5O1 44353043 IC50 = 7760 nM T76198 CQ1KR3 44353162 IC50 = 99000 nM T76198 C83VWP 44353167 IC50 = 160 nM T76198 CM60IB 44353169 IC50 = 1500 nM T76198 CZ9MS1 44353185 IC50 > 100000 nM T76198 C4LQZ7 44353186 IC50 = 1020 nM T76198 CTI2M5 44353269 IC50 = 10000 nM T76198 CPF3H9 44353282 IC50 = 1320 nM T76198 C8SFO0 44353289 IC50 > 100000 nM T76198 CWE72M 44353292 IC50 = 1480 nM T76198 C3DUQ8 44353300 IC50 = 2810 nM T76198 CY4OJ5 44353301 IC50 = 72300 nM T76198 CN0F5X 44353302 IC50 = 320 nM T76198 CJU36I 44353307 IC50 = 77600 nM T76198 CZLU91 44353309 IC50 = 17800 nM T76198 CS4B6M 44353316 IC50 = 47900 nM T76198 CH62KG 44353317 IC50 = 2880 nM T76198 C8GZV7 44353319 IC50 > 100000 nM T76198 C9CMY0 44364273 Ki = 16 nM T76198 CLN63A 44377464 Ki = 520 nM T76198 CMJ3B5 44385450 IC50 = 63000 nM T76198 CZ48UT 44385759 IC50 = 230000 nM T76198 C50TAM 44385825 IC50 = 5000 nM T76198 CR6D1I 44385826 IC50 = 700 nM T76198 CP79TX 44385934 IC50 = 1300 nM T76198 C3S8PG 44385988 IC50 = 10000 nM T76198 CJP2Y3 44386034 IC50 = 3800 nM T76198 C17OEZ 44386035 IC50 = 20000 nM T76198 C05CMA 44386125 IC50 = 5400 nM T76198 C3H9DS 44386126 IC50 = 700 nM T76198 CKNA65 44386134 IC50 = 38000 nM T76198 C20CKO 44386190 IC50 = 20000 nM T76198 CTX57O 44386253 IC50 = 86000 nM T76198 CY6ET8 44386321 IC50 = 1100 nM T76198 C38IEV 44386325 IC50 = 5500 nM T76198 C6HT0N 44386527 IC50 = 547000 nM T76198 CP3FJ5 44386678 IC50 = 25000 nM T76198 C3KA6N 44387045 IC50 = 72000 nM T76198 CR91XW 44387046 IC50 = 37000 nM T76198 C75WYL 44387118 IC50 = 13000 nM T76198 C87OVA 44387119 IC50 = 700 nM T76198 COR3J2 44387221 IC50 = 1000 nM T76198 CEJX46 44390242 Ki > 20000 nM T76198 C8EG2Q 44390268 Ki = 1500 nM T76198 C9MAN2 44390312 Ki > 20000 nM T76198 CDO76V 44390332 Ki > 20000 nM T76198 C0YXP5 44392456 Ki > 21000 nM T76198 CXB76Y 44392460 Ki = 140 nM T76198 CN1L7E 44392477 Ki = 200 nM T76198 C1YKS6 44392479 Ki > 21000 nM T76198 CP2O4K 44392512 Ki = 360 nM T76198 CI2KP5 44392527 Ki = 1200 nM T76198 CWL1X4 44400355 Ki > 1000 nM T76198 CSH9J2 44404954 Ki = 740 nM T76198 CJ1O3D 44411552 Ki = 100 nM T76198 C2UQV7 44411555 Ki = 180 nM T76198 CNM76B 44411567 Ki = 88 nM T76198 C69PSX 44411605 Ki = 330 nM T76198 CE3J1V 44411606 Ki = 1100 nM T76198 C7MCE5 44411635 Ki = 2700 nM T76198 C8ZUQ5 44411688 Ki = 5.1 nM T76198 C4AD5K 44411791 Ki = 6.6 nM T76198 CZ0X3F 44411797 Ki = 340 nM T76198 CUQ76I 44411798 Ki = 1800 nM T76198 CE49GA 44411799 Ki = 220 nM T76198 CLH8R3 44411809 Ki = 7.8 nM T76198 CH7UG4 44411813 Ki = 96 nM T76198 CRP5N3 44411814 Ki = 760 nM T76198 CCH0L3 44411851 Ki = 260 nM T76198 C5GD6H 44411889 Ki = 3700 nM T76198 CO41IV 44411890 Ki = 140 nM T76198 COMS38 44411896 Ki = 2100 nM T76198 C40QDV 44411984 Ki = 820 nM T76198 CIB2W5 44419347 Ki > 500 nM T76198 C91JXT 44419374 Ki > 500 nM T76198 CNF4W2 44419379 Ki > 500 nM T76198 C8KQP9 44448929 Ki = 79.43 nM T76198 C7N1IY 44448984 Ki = 398.11 nM T76198 C94ZPE 44448986 Ki = 31.62 nM T76198 C3E7YJ 44449112 Ki = 50.12 nM T76198 CXE43C 44450397 Ki = 310 nM T76198 CB2DC8 44450410 Ki = 286 nM T76198 C19SLD 44450427 Ki = 198 nM T76198 C8HA4B 44450496 Ki = 675 nM T76198 CDBE16 44450497 Ki = 7154 nM T76198 CH1O6B 44457567 IC50 = 440 nM T76198 CRB3C5 44457587 IC50 = 310 nM T76198 C4DL5C 44469677 IC50 > 10000 nM T76198 CVZW52 44537923 IC50 = 13700 nM T76198 CZY53M 44591457 Ki = 7 nM T76198 CJUX12 44591458 Ki = 2917 nM T76198 C5ZRQ7 44591477 Ki > 20000 nM T76198 CFI4O5 44591512 Ki = 687 nM T76198 C87ZCK 44591513 Ki = 1687 nM T76198 CH2W6M 44591514 Ki = 990 nM T76198 CI5SP2 44591515 Ki = 415 nM T76198 COH31P 44591516 Ki = 587 nM T76198 CH7LE5 44591535 Ki = 3428 nM T76198 CZ2UO0 44591536 Ki = 626 nM T76198 C4DJH3 44591537 Ki = 468 nM T76198 CF5O6R 44591561 Ki > 20000 nM T76198 CMZ6B3 44591562 Ki = 6144 nM T76198 C6Z2MX 44591563 Ki = 186 nM T76198 CD9KX4 44591762 Ki = 41.5 nM T76198 CJ6S7Q 44591806 Ki = 339.8 nM T76198 CT0L2W 44591807 Ki = 13.9 nM T76198 CRA6S0 45109984 Ki > 22000 nM T76198 C3JE7N 45109987 Ki > 21000 nM T76198 CA28PL 45109988 Ki > 7200 nM T76198 CN6P8B 45109989 Ki > 7200 nM T76198 CY2BK4 45110108 Ki > 7200 nM T76198 CR1KP4 45110109 Ki > 7200 nM T76198 CR6UW4 45112038 Ki > 71000 nM T76198 CB5O6V 45269307 IC50 > 100000 nM T76198 C03ETI 45270148 IC50 > 100000 nM T76198 CY70SI 45270983 IC50 > 100000 nM T76198 C2XH3A 45270987 IC50 > 100000 nM T76198 C35DUQ 45272700 IC50 > 100000 nM T76198 CKUI32 45272704 IC50 > 100000 nM T76198 C3U7KT 45273637 Ki > 7000 nM T76198 CA4LM0 46890179 Ki = 7800 nM T76198 CZ6OK4 46890180 Ki = 3400 nM T76198 C0A2CI 46890616 Ki >= 504 nM T76198 CW52VH 46890658 Ki >= 260 nM T76198 CXQ2W0 46890659 Ki >= 580 nM T76198 CQ20RC 46890660 Ki >= 100 nM T76198 CM06FG 50898361 Ki = 61 nM T76198 CZ9UD6 50901657 IC50 > 100000 nM T76198 C8VNM2 51003549 Ki > 22000 nM T76198 CJD25G 52920263 IC50 = 560000 nM T76198 C3XYP8 52941281 Ki = 362 nM T76198 C6SPT4 52943623 Ki = 112 nM T76198 CE04FW 52944928 Ki = 100 nM T76198 CA41UT 52944959 Ki = 93 nM T76198 CX8L6T 52945002 Ki = 1481 nM T76198 C4K6BH 52946883 Ki > 10000 nM T76198 C9WUH5 52948543 Ki = 270 nM T76198 CI8TP9 52948585 Ki = 292 nM T76198 CK9DR7 52949846 Ki = 106 nM T76198 CTU93P 53316532 Ki > 6800 nM T76198 C4P2CV 53316653 Ki > 7139 nM T76198 CS4G5H 53316671 Ki = 719 nM T76198 CL96IZ 53316672 Ki > 5591 nM T76198 CBT1P4 53316673 Ki > 7181 nM T76198 C8D7UQ 53317569 Ki = 1840 nM T76198 C1CFU7 53317642 Ki > 7054 nM T76198 CXV3W2 53317718 Ki = 1569 nM T76198 C0ZH3X 53317854 Ki > 6800 nM T76198 CP14EK 53317957 Ki = 727 nM T76198 C97LDX 53317958 Ki = 3949 nM T76198 C5WO9J 53317977 Ki > 7054 nM T76198 COJ82D 53319320 Ki = 962 nM T76198 C4T9BV 53319321 Ki = 2142 nM T76198 CE86AP 53319322 Ki > 7096 nM T76198 CV8M5K 53320594 Ki > 21660 nM T76198 CZL85A 53320595 Ki = 1872 nM T76198 C8EO2U 53320616 Ki = 2890 nM T76198 C5HY9K 53320617 Ki = 904 nM T76198 CZ40CV 53320618 Ki = 2840 nM T76198 CIU6E0 53321678 Ki > 5591 nM T76198 C7D5BN 53321784 Ki > 22000 nM T76198 C5QOI8 53321785 Ki > 27000 nM T76198 C89DLV 53321923 Ki = 1330 nM T76198 C29QNI 53321924 Ki = 1039 nM T76198 CJ7C4U 53321925 Ki > 5745 nM T76198 CB5S0H 53322785 Ki = 1357 nM T76198 CPI3O6 53323246 Ki = 888 nM T76198 C2KRB3 53323266 Ki = 427 nM T76198 CMK0A1 53323267 Ki = 10.9 nM T76198 C4ZP8Y 53323268 Ki = 1222 nM T76198 CTOY32 53324111 Ki = 2118 nM T76198 CE23YH 53324462 Ki > 1000 nM T76198 CF9SZ3 53324589 Ki = 1518 nM T76198 CUS37X 53325907 Ki > 7247 nM T76198 CZ1SE0 53325908 Ki = 2152 nM T76198 CH8S3T 53325909 Ki > 21160 nM T76198 C9DR3V 53325910 Ki > 7054 nM T76198 CZ7WN5 53325911 Ki > 5591 nM T76198 CEMU31 53325912 Ki > 7181 nM T76198 CAL29U 53326879 Ki > 6489 nM T76198 CZ9D6X 53358921 IC50 = 7600 nM T76198 COFI65 53358922 IC50 > 10000 nM T76198 CY40UL 53494965 Ki > 10000 nM T76198 C9HK6G 54582728 Ki > 1000 nM T76198 C2RJM1 54583706 Ki > 1000 nM T76198 CRS92B 54592351 IC50 = 1500 nM T76198 CKHP37 54669850 IC50 = 198 nM T76198 CO6V5Y 54757768 IC50 > 10000 nM T76198 COKJ36 54757769 IC50 = 3801 nM T76198 CCMS10 54757770 IC50 = 5303 nM T76198 C68TXA 54757771 IC50 = 21853 nM T76198 CZ12NO 54757965 IC50 = 15117 nM T76198 C6AVP5 54758053 IC50 = 64 nM T76198 CYE26R 54758054 IC50 = 377 nM T76198 C5YX0Z 56659855 IC50 = 38000 nM T76198 CR4U7M 56665068 Ki > 10000 nM T76198 CWR1Z7 56665984 Ki > 13000 nM T76198 C4AOU2 56672019 Ki > 10000 nM T76198 C4ZE6P 56672020 Ki > 10000 nM T76198 CH3R8E 56675398 Ki > 10000 nM T76198 CU7K0N 56680341 IC50 = 39000 nM T76198 C6T5SC 56680464 IC50 = 41 nM T76198 C1U7XJ 56924869 IC50 = 62400 nM T76198 C37SMZ 57505249 IC50 > 1000 nM T76198 C0U1HA 59179260 IC50 = 200 nM T76198 CVM9Q1 68503758 IC50 > 25000 nM T76198 CA15ND 68505312 IC50 > 25000 nM T76198 C0US2T 68505327 IC50 > 25000 nM T76198 CX8W7F 68508048 IC50 > 25000 nM T76198 COJ4Q1 69315206 IC50 > 25000 nM T76198 C9KGN4 70684971 IC50 = 510 nM T76198 C6JI0C 70685025 IC50 = 5700 nM T76198 COI75G 71138349 IC50 = 54 nM T76198 C7LC9G 71138378 IC50 = 892 nM T76198 C86ATI 71138563 IC50 = 59 nM T76198 CV28YI 71450058 Ki = 740 nM T76198 CLMR38 71450832 IC50 = 1400 nM T76198 C6OQ3R 71451008 IC50 = 77 nM T76198 CXP2S8 71456310 IC50 = 105 nM T76198 CDT62N 71460870 Ki = 15 nM T76198 C8XJ0I 71733818 IC50 > 25000 nM T76198 CXC78L 71733909 IC50 > 25000 nM T76198 C7B5XE 71733910 IC50 > 25000 nM T76198 CQ21ZD 71733911 IC50 > 25000 nM T76198 CZG0S2 71733912 IC50 > 25000 nM T76198 CQ1YL7 71740056 IC50 = 6130 nM T76198 C6WM8U 71740057 IC50 = 1470 nM T76198 CU5YE0 71740179 IC50 = 1780 nM T76198 CLV21C 71740180 IC50 = 2380 nM T76198 CTXJ20 71740181 IC50 = 690 nM T76198 C8CD1Y 71740182 IC50 = 680 nM T76198 CEZW12 71740183 IC50 = 1350 nM T76198 C6RAL4 71740184 IC50 = 680 nM T76198 CZLG08 71740185 IC50 = 900 nM T76198 CUM73W 71740307 IC50 = 9620 nM T76198 CO64BZ 71740308 IC50 = 3890 nM T76198 CC8ZW0 71740309 IC50 = 9430 nM T76198 COL4H5 71740310 IC50 = 8490 nM T76198 CG51CP 71740311 IC50 = 5270 nM T76198 CVH56F 71740312 IC50 = 8640 nM T76198 CYIG30 71740313 IC50 = 9470 nM T76198 CJA0S2 71740438 IC50 = 5310 nM T76198 CC7T9Q 71740439 IC50 = 8520 nM T76198 C49ZPM 71740440 IC50 = 9490 nM T76198 C4UF0I 71740441 IC50 = 5520 nM T76198 C9VKG5 71740442 IC50 = 9490 nM T76198 C03BRA 71740443 IC50 = 10120 nM T76198 CEIT37 71740444 IC50 = 2750 nM T76198 C5SA6C 71740557 IC50 = 3190 nM T76198 CXD2L6 71740558 IC50 = 9110 nM T76198 CAPE23 71740559 IC50 = 1590 nM T76198 CC1R3F 71740560 IC50 = 2950 nM T76198 CFM60J 71740561 IC50 = 4220 nM T76198 C69ETO 71740562 IC50 = 1040 nM T76198 CP93IL 71740563 IC50 = 1040 nM T76198 C6AU5T 71740667 IC50 = 7830 nM T76198 CUP17N 71740668 IC50 = 4640 nM T76198 C25DJX 71740669 IC50 = 6450 nM T76198 CUAW76 73354171 IC50 = 35.8 nM T76198 C6W5KZ 117630015 IC50 = 2760 nM T76198 CW75AE 117630458 IC50 = 29.2 nM T76198 CS02NG 117630548 IC50 = 3.9 nM T76198 C86OSM 117630978 IC50 = 0.015 nM T76198 C7RIV2 117631017 IC50 = 11.2 nM T76198 C9H8LF 117631097 IC50 = 6.5 nM T76198 C4EF6U 117631354 IC50 = 0.052 nM T76198 CGCA83 118711723 IC50 = 1140 nM T76198 CV37QW 118714499 IC50 = 10.7 nM T76198 CT8O1N 118714500 IC50 = 891 nM T76198 CUV5Y0 118715454 EC50 > 30000 nM T76198 CC0HS2 118718127 IC50 = 115000 nM T76198 CTQ20K 118719206 IC50 = 3800 nM T76198 CZ24FT 122197353 IC50 = 2000 nM T76198 CWXR72 127029417 Ki > 50000 nM T76198 CJAQ90 127047381 Ki > 50000 nM T76198 CND51M 135528684 Ki = 120226.44 nM T76198 C3KQ6B 19701789 IC50 = 50 nM T76198 CQ9K6L 19701795 IC50 = 20 nM T76198 C3WD4X 19701804 IC50 = 580 nM T76198 CR2U5D 44304263 IC50 = 60 nM T76198 CHL94N 44304279 IC50 = 1700 nM T76198 CJT8H2 44304290 IC50 = 190 nM T76198 C6I7EB 44304362 IC50 = 20 nM T76198 CKJ70Q 44304533 IC50 = 520 nM T76198 D02MXT 24952929 Ki > 6800 nM T76198 D03OYD 5311240 EC50 = 8000 nM T76198 D03PLH 5311493 Ki = 5.5 nM T76198 D07UDT 15551229 Ki > 500 nM T76198 D08KZJ 11384493 Ki = 1394 nM T76198 D0O9ES 5311053 EC50 = 2400 nM T76198 D0QH5C 230826 Ki > 10000 nM T76198 D0S2LO 9864831 Ki > 13000 nM T76198 D0S6NE 11306423 Ki = 220 nM T76198 D0TA0L 23685469 Ki > 1000 nM T76198 D0WV5J 44450494 Ki = 17 nM T76198 D0X5MA 5311175 IC50 = 50 nM T76198 D0XB3U 5312142 IC50 = 53.1 nM T76198 D0Y1IF 23664784 Ki > 1000 nM T76198 D0Z3XJ 9817405 Ki > 500 nM T68547 D00SQN 12136798 IC50 = 167 nM T68547 D01QIN 60823 IC50 = 11619 nM T68547 D03RTS 2662 IC50 = 1185 nM T68547 D06WTZ 53232 IC50 = 11911 nM T68547 D07POC 176870 IC50 > 32000 nM T68547 D08CDI 208908 IC50 > 10000 nM T68547 D09DHY 6167 IC50 > 20 ug.mL-1 T68547 D0AZ3C 5291 IC50 > 100000 nM T68547 D0B7EB 36462 IC50 > 20 ug.mL-1 T68547 D0E3SH 6918837 Ki = 0.54 nM T68547 D0E7PQ 5311 Ki = 1.3 nM T68547 D0L7LC 5352062 Ki = 0.0015 nM T68547 D0R9BG 1990 IC50 = 625000 nM T68547 D0Y3KG 3121 IC50 = 39000 nM T68547 D00FHR 9865515 Ki = 9 nM T68547 D00SSZ 11178958 IC50 = 3.3 nM T68547 D01WKZ 53340426 IC50 = 35 nM T68547 D05KED 53340666 IC50 = 38 nM T68547 D06TKI 49857317 IC50 = 3 nM T68547 D07FPY 6918877 Ki = 11 nM T68547 D09XIZ 11538455 Ki = 0.03 nM T68547 D0B3FV 6445533 Ki = 0.55 nM T68547 D0B7CH 4775 IC50 = 64000 nM T68547 D0E6UZ 54575456 IC50 = 0.36 nM T68547 D0GE5B 56654642 Ki = 32 nM T68547 D0GH3Q 9804992 Ki = 2 nM T68547 D0L2UQ 49855250 Ki = 16 nM T68547 D0M8FD 4261 Ki = 22 nM T68547 D0V0SL 11749858 Ki = 7 nM T68547 D0VE1W 6918876 IC50 = 52 nM T68547 D0XT6W 6918638 Ki = 0.85 nM T68547 D0Z4RC 24756910 IC50 = 4.5 nM T68547 D03SZR 5353484 IC50 = 10 nM T68547 D0J8OC 5186 Ki = 1.5 nM T68547 D00HXJ 118884610 Ki = 358 nM T68547 D00OWF 5280953 IC50 > 1000 nM T68547 D0CH8Q 56965342 IC50 = 4800 nM T68547 D0JY1I 42613483 IC50 = 80 nM T68547 D0L1NO 72722126 IC50 = 14000 nM T68547 D0N2DK 72710871 IC50 = 2 nM T68547 D0Q1QY 57381425 IC50 = 94 nM T68547 D0QX3G 71532921 IC50 = 2100 nM T68547 D0V5IQ 130227480 IC50 = 187 nM T68547 D0YN2T 86302836 IC50 > 50000 nM T68547 D0ZG5X 71811260 IC50 = 1050 nM T68547 D0N3SH 4996 Ki = 2.7 nM T68547 D0W9NH 2746 Ki = 50 nM T68547 C8HA6K 3994 IC50 = 2960 nM T68547 CCK23B 4144 IC50 = 100 nM T68547 CI7J6E 4148 IC50 = 4.5 nM T68547 C5S2BK 5048 IC50 = 2000 nM T68547 CBIR94 10313 IC50 = 4730 nM T68547 C03POM 28115 IC50 < 20 nM T68547 CL25FN 76175 IC50 > 30000 nM T68547 C4O1AZ 79419 IC50 = 4800 nM T68547 C1N2KZ 88129 IC50 = 560000 nM T68547 C5Z1QA 96028 IC50 > 200000 nM T68547 CE42TU 119411 IC50 > 25000 nM T68547 CW70DI 211808 IC50 = 50000 nM T68547 CP62UE 239511 IC50 = 6600 nM T68547 CH1JD3 419176 IC50 = 7000 nM T68547 C0Y4WC 614947 Ki > 2500 nM T68547 C0EM9B 801008 IC50 = 19400 nM T68547 CBC31X 817096 IC50 = 2454.71 nM T68547 CU3HS2 1108280 IC50 > 100000 nM T68547 C96GFC 1798422 IC50 = 129200 nM T68547 C94IXC 2173124 IC50 = 4060 nM T68547 C58NGX 2175719 IC50 = 4050 nM T68547 CJCY71 2295078 IC50 = 1730 nM T68547 CG41FO 2423676 IC50 = 3310 nM T68547 CEO31B 2423687 IC50 = 3650 nM T68547 CA9TW1 2723947 IC50 < 20 nM T68547 CQ6TG1 2803102 IC50 > 10000 nM T68547 CSH3B1 3042223 IC50 > 50000 nM T68547 CN4M6D 5281220 IC50 = 38000 nM T68547 C7KAR5 5353765 IC50 = 10 nM T68547 CH5FO1 5353767 IC50 = 200 nM T68547 CT68UM 5353768 IC50 = 2000 nM T68547 CXUP49 5353769 IC50 = 600 nM T68547 C7RZA4 5353770 IC50 = 90 nM T68547 CSIJ53 5793932 IC50 = 11400 nM T68547 C18ENP 6918846 Ki = 12 nM T68547 C1RD7E 6918878 Ki < 0.2 nM T68547 CE9LP2 9543539 IC50 = 199 nM T68547 CJ07ZA 9800555 IC50 = 95 nM T68547 C1OD4S 9804482 IC50 = 2.5 nM T68547 CAU23Y 9806551 IC50 = 0.4 nM T68547 CPE85S 9824191 IC50 = 2000 nM T68547 CX5W3K 9824244 IC50 = 9.4 nM T68547 CC0EU7 9828788 IC50 = 1.6 nM T68547 CLYJ85 9848223 IC50 = 180 nM T68547 C25KPR 9856090 IC50 = 67000 nM T68547 C4GBE9 9860473 IC50 = 100 nM T68547 CH2KP3 9864818 IC50 = 12.1 nM T68547 C8M4KZ 9866917 IC50 = 130 nM T68547 CPS24V 9880847 IC50 = 15 nM T68547 C0MG5Q 9887245 IC50 = 2000 nM T68547 CEG83X 9889124 IC50 = 3.5 nM T68547 CSW4Y1 9891541 IC50 = 160 nM T68547 CQ82UG 9923301 IC50 = 500 nM T68547 C81EYJ 9923508 IC50 = 3.2 nM T68547 CQG4V8 9924543 IC50 = 1.6 nM T68547 C1Y4EK 9924842 IC50 = 100 nM T68547 CX0FB5 9931544 IC50 = 18 nM T68547 CE7M4R 9953205 IC50 = 3000 nM T68547 CO03VC 9956086 IC50 = 14.5 nM T68547 C49KZT 9968179 IC50 = 4000 nM T68547 CI21BO 9976852 IC50 = 6 nM T68547 C4J6YE 9977875 IC50 = 7 nM T68547 C8VSK1 9978533 IC50 = 2 nM T68547 CDT7U0 9998313 IC50 = 63 nM T68547 CR98AV 9999602 IC50 = 160 nM T68547 CR9ZD0 10004160 IC50 = 50 nM T68547 CZL7C8 10017099 IC50 = 6 nM T68547 C3GCS5 10044793 IC50 = 3000 nM T68547 CY76FQ 10059360 IC50 = 186 nM T68547 CXA5J1 10068980 IC50 = 20 nM T68547 CVC3A9 10071120 IC50 = 1220 nM T68547 CCD3S6 10090483 IC50 = 50 nM T68547 C5R3EY 10091222 IC50 = 12 nM T68547 CM9UQ1 10109962 IC50 = 2000 nM T68547 CQDG65 10110195 IC50 = 300 nM T68547 CTBY37 10111144 EC50 = 1000 nM T68547 C24BEW 10112461 IC50 = 200 nM T68547 CKX3I1 10114795 IC50 = 50 nM T68547 CUT8Y9 10117759 IC50 = 400 nM T68547 CW1K6E 10133863 IC50 = 90 nM T68547 CWA9R2 10135838 IC50 = 11 nM T68547 CL4C9H 10154438 Ki = 1.3 nM T68547 C4HLA0 10157327 IC50 = 60 nM T68547 CR1G8D 10157889 IC50 = 3000 nM T68547 CWV5F1 10161509 IC50 = 300 nM T68547 CWPN64 10177542 IC50 = 200 nM T68547 CIZ05J 10179372 IC50 = 70 nM T68547 CC5WG3 10193406 IC50 = 123.03 nM T68547 CP34BN 10201125 IC50 = 80 nM T68547 C4AQ7F 10201496 IC50 = 5000 nM T68547 C6YX1B 10202306 IC50 = 300 nM T68547 C81YFS 10204219 IC50 = 1000 nM T68547 C0HAW1 10223095 IC50 = 3000 nM T68547 C6O0YK 10226045 IC50 = 4000 nM T68547 CCA69X 10229117 IC50 = 100 nM T68547 CON61Q 10246764 IC50 = 21 nM T68547 CY2CR9 10246779 IC50 = 33 nM T68547 CU4E9S 10247137 IC50 = 60 nM T68547 CB2OV7 10266393 IC50 = 120 nM T68547 C82BPN 10269384 IC50 = 2000 nM T68547 CO6X0M 10270022 IC50 = 3000 nM T68547 C5DMV1 10270750 IC50 = 200 nM T68547 CKA1O3 10271347 IC50 = 80 nM T68547 CCW2X7 10271530 IC50 = 100 nM T68547 CK3I9Y 10271952 IC50 = 40 nM T68547 C9ZAH0 10273460 IC50 = 5000 nM T68547 CH1AX8 10278510 IC50 = 800 nM T68547 CB28EY 10292566 IC50 = 30 nM T68547 C1KH8L 10293869 IC50 = 100 nM T68547 CUB5K3 10296337 IC50 = 300 nM T68547 C5VF2H 10298829 IC50 = 1000 nM T68547 CZ8M6A 10300469 IC50 = 70 nM T68547 C7RC1E 10309899 IC50 = 2.5 nM T68547 C5S8XH 10340474 IC50 = 50 nM T68547 CP5D1Y 10341900 IC50 = 1000 nM T68547 CSZ54R 10342304 IC50 = 1000 nM T68547 C1G9YS 10362929 IC50 = 50 nM T68547 CN5IT3 10381402 IC50 = 79 nM T68547 CMX76Q 10388312 IC50 = 1500 nM T68547 CYB45J 10436141 EC50 = 1000 nM T68547 C9G8LC 10450420 IC50 = 100 nM T68547 CG0D6N 10451940 IC50 > 100000 nM T68547 C9OU5F 10464879 Ki > 2500 nM T68547 CY9I0S 10470023 IC50 = 153 nM T68547 CDY91S 10584105 Ki > 2500 nM T68547 CE8H0J 10602086 IC50 = 3600 nM T68547 C3KT5X 10707192 IC50 = 1380 nM T68547 CSMT47 10728039 Ki > 2500 nM T68547 C3FC7X 10800939 IC50 = 21200 nM T68547 COU1F3 10861784 IC50 > 25000 nM T68547 C7PL3U 10872455 IC50 = 100 nM T68547 C5FB6Z 10873314 IC50 = 200 nM T68547 C7KEN0 10874340 IC50 = 1000 nM T68547 C80ZXG 10881097 IC50 = 5 nM T68547 C6IY9G 10884912 IC50 = 3000 nM T68547 CE68AK 10906789 IC50 = 4000 nM T68547 CXEA43 10914552 IC50 = 200 nM T68547 CQ0H2D 10916552 IC50 = 2000 nM T68547 C1XZ0F 10928759 IC50 = 9000 nM T68547 CB06IG 10961225 IC50 = 3000 nM T68547 CEOQ09 10972684 IC50 = 3000 nM T68547 C17HLX 10990261 IC50 = 3000 nM T68547 C3O6IV 10992230 IC50 = 50 nM T68547 CW79IF 11001628 IC50 = 45 nM T68547 C07BVO 11003161 IC50 = 500 nM T68547 CB54GF 11004935 IC50 > 25000 nM T68547 CK8UV7 11019840 Ki > 2500 nM T68547 CU64OX 11024075 IC50 = 9.5 nM T68547 C1H9RC 11036226 IC50 = 50 nM T68547 C3PC7D 11056092 IC50 = 600 nM T68547 CHBS32 11068279 IC50 = 1000 nM T68547 CEPM03 11068867 IC50 = 23 nM T68547 C5KRO7 11112665 IC50 = 1000 nM T68547 CR8LU2 11118652 IC50 = 50 nM T68547 CQ6ZE8 11153178 IC50 = 2300 nM T68547 CI0S5H 11153574 IC50 = 190 nM T68547 C5B4OC 11153716 IC50 = 1200 nM T68547 CZV67X 11155508 IC50 = 7.7 nM T68547 CFW0R5 11164133 IC50 = 20 nM T68547 CW2GJ0 11166750 IC50 = 10 nM T68547 C5P3EI 11167060 IC50 = 50 nM T68547 CE0U4M 11176541 IC50 = 355 nM T68547 CFEN82 11177718 IC50 = 79 nM T68547 C5JR3Q 11184660 IC50 > 10000 nM T68547 C4H3CU 11188147 IC50 = 80 nM T68547 CMQ38G 11199235 IC50 = 79 nM T68547 CA48NR 11199635 IC50 > 100 nM T68547 C14EJI 11201165 IC50 = 48 nM T68547 CX71WU 11202558 IC50 = 54 nM T68547 C5SEQ1 11202590 IC50 = 47 nM T68547 CT1W4H 11210084 IC50 = 1900 nM T68547 C8G5WP 11210533 IC50 = 8800 nM T68547 CBVT14 11212063 IC50 = 880 nM T68547 CG27ZR 11212396 IC50 = 7.9 nM T68547 C1OPI2 11222757 IC50 = 170 nM T68547 CCJ97D 11223267 IC50 = 250 nM T68547 C89SVA 11223999 IC50 = 5 nM T68547 CVC05Z 11233783 IC50 = 140 nM T68547 CTQ76N 11235378 IC50 = 160 nM T68547 CYJ60V 11244651 IC50 = 25600 nM T68547 C6TX9W 11255848 IC50 = 11.5 nM T68547 CSO06H 11259022 IC50 = 10 nM T68547 CI7W3O 11267278 IC50 = 1080 nM T68547 CG4BO7 11267357 IC50 = 31 nM T68547 C6AKW1 11270791 IC50 = 12 nM T68547 CM6ZW2 11279156 IC50 = 1430 nM T68547 C1W6IV 11302939 IC50 = 41 nM T68547 CEH69P 11315473 IC50 = 93 nM T68547 CHAZ68 11316470 IC50 = 250 nM T68547 CI95SE 11318367 IC50 = 1 nM T68547 CV9Y4T 11326181 IC50 = 31 nM T68547 CBY0U5 11326448 IC50 = 210 nM T68547 C82EFX 11326996 IC50 = 555 nM T68547 C0WDK4 11327236 IC50 = 160 nM T68547 CI3DO1 11339463 IC50 = 200 nM T68547 CCT25X 11340446 IC50 = 48 nM T68547 CAM46F 11347217 IC50 = 1700 nM T68547 C0BQ6D 11348476 IC50 = 3200 nM T68547 CS2N4U 11350045 IC50 = 26 nM T68547 C3R8PT 11359017 IC50 = 100 nM T68547 CQIG34 11359309 IC50 = 10 nM T68547 CDL0O2 11359758 IC50 = 55 nM T68547 CZT79Q 11360420 IC50 = 7.9 nM T68547 C46EZD 11382208 IC50 = 3300 nM T68547 CU96OI 11383207 IC50 = 530 nM T68547 C28ZES 11385344 IC50 = 51.3 nM T68547 CY34EQ 11393847 IC50 = 60 nM T68547 C9QB0C 11396478 IC50 = 7.9 nM T68547 CCYJ34 11404457 IC50 = 260 nM T68547 C0LO5S 11418079 IC50 = 410 nM T68547 CA92KL 11420425 IC50 = 170 nM T68547 CGU10B 11428430 IC50 = 79 nM T68547 CJD61L 11428534 IC50 = 170 nM T68547 CVH8N1 11430412 IC50 = 31 nM T68547 CRTV86 11430535 IC50 = 40 nM T68547 CDAT72 11433190 IC50 > 100000 nM T68547 CKB54N 11438800 IC50 = 200 nM T68547 CNU8D3 11438971 EC50 = 12000 nM T68547 C2V7HJ 11439694 IC50 = 36 nM T68547 C5HP1B 11441977 IC50 = 5 nM T68547 CI9AG3 11449652 IC50 = 170 nM T68547 CLJ27W 11449785 IC50 = 203.5 nM T68547 CMB9R2 11452638 IC50 = 392 nM T68547 C49NIT 11452842 IC50 = 310 nM T68547 C7Z8NH 11454564 IC50 = 42 nM T68547 C8PQ2H 11461110 IC50 = 106.5 nM T68547 CW9AB4 11473538 IC50 = 170 nM T68547 C3BGS1 11473639 EC50 = 1500 nM T68547 CLW8E4 11477101 IC50 = 21 nM T68547 CJ7W4K 11478458 IC50 = 9.5 nM T68547 CASI20 11485016 IC50 = 40 nM T68547 C9UY7W 11486323 IC50 = 1600 nM T68547 CS74ML 11508879 IC50 = 4600 nM T68547 C0L4FB 11512777 IC50 = 730 nM T68547 CJGL17 11539751 IC50 = 10.47 nM T68547 C5JEZ9 11544171 IC50 = 12.3 nM T68547 CRZ7H2 11556677 IC50 = 13 nM T68547 C2F9NT 11558827 IC50 = 209 nM T68547 C86YFM 11575878 IC50 = 19.05 nM T68547 CR75XL 11578056 IC50 = 220 nM T68547 C5JBF8 11589054 IC50 = 9.772 nM T68547 C7A3OZ 11590444 IC50 = 33.11 nM T68547 C3LO6F 11597868 IC50 = 13.18 nM T68547 C96ZFI 11599797 IC50 = 150 nM T68547 C8GVH9 11603554 IC50 = 18.62 nM T68547 C0FI7A 11603622 IC50 = 110 nM T68547 C1EJO5 11610262 IC50 = 45 nM T68547 C9UI2V 11617038 IC50 = 16 nM T68547 CA6X1R 11619076 IC50 = 9.772 nM T68547 CB3U6H 11628528 IC50 = 162 nM T68547 CWE63G 11633344 IC50 = 18.62 nM T68547 CK9SY1 11635398 IC50 = 220 nM T68547 C3DXH7 11638904 IC50 = 38.02 nM T68547 CHR61G 11640784 IC50 = 250 nM T68547 C24SBP 11657529 IC50 = 30 nM T68547 CP4V9X 11664428 IC50 = 1760 nM T68547 CQ32FV 11664499 IC50 = 0.8 nM T68547 CD9XU6 11675152 IC50 = 21.38 nM T68547 CG9OC4 11682502 IC50 = 7.1 nM T68547 C2JSO8 11683474 IC50 = 38.02 nM T68547 CYB26W 11688197 IC50 = 605 nM T68547 CJ2UA0 11690271 IC50 = 1170 nM T68547 CCF7Y4 11696355 IC50 = 11 nM T68547 CC3GQ0 11700059 IC50 = 26 nM T68547 CK1FB9 11710573 IC50 = 50.12 nM T68547 C9WI7N 11712071 IC50 = 16.22 nM T68547 CX2GR8 11723098 IC50 = 100 nM T68547 C8N9UZ 11724319 IC50 = 300 nM T68547 CL4UP0 11739171 IC50 = 220 nM T68547 CNDE90 11772176 IC50 = 70 nM T68547 CKRA48 11772295 IC50 = 20 nM T68547 CGE0C3 11774481 IC50 = 270 nM T68547 CE4Z0Y 11844891 IC50 = 1210 nM T68547 C6JF9E 11844892 IC50 = 1270 nM T68547 CY0WV6 11844893 IC50 = 900 nM T68547 CU0M1E 11947684 IC50 = 2.4 nM T68547 CF06BI 11963978 IC50 = 1.6 nM T68547 C9G1BN 11993595 IC50 = 4800 nM T68547 CH5JS7 11993694 IC50 = 83 nM T68547 CJQ8L0 12001305 IC50 = 1.6 nM T68547 C1BVY9 12325934 IC50 > 30000 nM T68547 CKI97Z 12344252 IC50 > 200000 nM T68547 CKSL53 12507616 IC50 > 200000 nM T68547 CJ94OC 12542182 Ki > 2500 nM T68547 COF8W3 13008156 IC50 > 50000 nM T68547 C06UTF 13507024 IC50 = 11 nM T68547 CA07QT 13873842 IC50 = 220 nM T68547 C4XJ8M 13889849 Ki = 190 nM T68547 C1KR4L 14113324 IC50 > 50000 nM T68547 C15MQN 14113325 IC50 > 50000 nM T68547 C1D0WF 14362924 Ki > 12500000 nM T68547 C2D1KP 15983982 Ki = 19 nM T68547 CA2YF9 15984018 IC50 = 320 nM T68547 C7DK5L 15984110 IC50 = 440 nM T68547 CHB82E 15986417 IC50 > 100000 nM T68547 C52EVH 15986418 IC50 = 5510 nM T68547 CS1QO9 15986509 IC50 = 8550 nM T68547 CC4BR6 16005382 IC50 = 34 nM T68547 CLG89X 16005547 IC50 = 229 nM T68547 C0BNE7 16005851 IC50 = 47 nM T68547 C2CHS1 16005949 IC50 = 200 nM T68547 CQ2LP3 16006351 IC50 = 7195 nM T68547 C8PBI9 16006352 IC50 = 196 nM T68547 C5T1WF 16006672 IC50 = 36 nM T68547 CWEZ01 16006673 IC50 = 199 nM T68547 CI53QT 16006776 IC50 = 103 nM T68547 C24RQO 16006779 IC50 = 35 nM T68547 C13DCE 16006876 IC50 = 21 nM T68547 C3JDK5 16006877 IC50 = 63 nM T68547 C7ZOV4 16006878 IC50 = 56 nM T68547 CQGC05 16036765 IC50 = 55 nM T68547 CM3T2E 16049824 IC50 = 11 nM T68547 CRL96K 16065840 IC50 = 550 nM T68547 C30UFT 16066811 IC50 = 79 nM T68547 CFK8J5 16068056 Ki = 24 nM T68547 C37TQE 16068057 IC50 = 308 nM T68547 CBG52I 16068168 IC50 = 150 nM T68547 CP1R3O 16068171 IC50 = 175 nM T68547 C4U0QY 16068175 IC50 = 135 nM T68547 CRH0O8 16068287 IC50 = 45 nM T68547 CZDK28 16068489 IC50 = 23 nM T68547 CU3GD2 16068491 IC50 = 155 nM T68547 C9YHZ8 16068492 IC50 = 335 nM T68547 CJN9P6 16068493 IC50 = 77 nM T68547 CMQP70 16068495 Ki = 26 nM T68547 CZC63A 16068590 IC50 = 165 nM T68547 CT84XO 16068594 Ki = 20 nM T68547 CF3ZG5 16068595 Ki = 11 nM T68547 CQ1XJ8 16068694 IC50 = 90 nM T68547 CDAB64 16068801 IC50 = 27 nM T68547 CJ4PG2 16068802 IC50 = 110 nM T68547 C4C1BT 16068803 IC50 = 68 nM T68547 CL60CA 16068912 Ki = 10 nM T68547 CXDH36 16068915 IC50 = 29 nM T68547 CO4L6G 16068916 IC50 = 41 nM T68547 CVG39Y 16068917 IC50 = 15 nM T68547 CO8MV2 16068918 IC50 = 22 nM T68547 CS9MH1 16068919 IC50 = 45 nM T68547 C4FYH5 16069015 IC50 = 41 nM T68547 CQ6TH9 16069016 IC50 = 41 nM T68547 C0NT1R 16069017 IC50 = 125 nM T68547 C6UL1O 16069018 IC50 = 190 nM T68547 CQX71L 16069019 IC50 = 105 nM T68547 COY6R8 16069021 IC50 = 109 nM T68547 CVO73I 16069022 IC50 = 158 nM T68547 CVT0E7 16070046 IC50 = 39 nM T68547 C9ZQB3 16095102 Ki > 5000 nM T68547 C80XYC 16095113 Ki > 5000 nM T68547 C6RE2F 16220721 Ki = 4.15 nM T68547 C09FZM 16220753 IC50 = 174 nM T68547 CJR3T1 16658996 IC50 = 530 nM T68547 CFLC70 16659045 IC50 = 1880 nM T68547 C82FSW 16662634 IC50 = 40 nM T68547 CCB25E 16662685 IC50 = 435 nM T68547 CH7B0D 16662686 IC50 = 582 nM T68547 CYX28Q 16662687 IC50 = 255 nM T68547 CYV15U 16662688 IC50 = 304 nM T68547 CMV50K 16662689 IC50 = 326 nM T68547 CAF87C 16662690 IC50 = 242 nM T68547 C2VJ8S 16662752 IC50 = 301 nM T68547 C8GQ7N 16662753 IC50 = 352 nM T68547 C1BCK7 16662754 IC50 = 821 nM T68547 CDO65G 16662755 IC50 = 140 nM T68547 CRN51J 16662757 IC50 = 77 nM T68547 CSMJ63 16662758 IC50 = 588 nM T68547 CHTP71 16662806 IC50 = 169 nM T68547 CLZG05 16662808 IC50 = 149 nM T68547 CH9TC5 16662811 IC50 = 529 nM T68547 C4MES5 16662813 IC50 = 39 nM T68547 C72CVD 16662872 IC50 = 75 nM T68547 C8TRL4 16662873 IC50 = 47 nM T68547 C4ZU7Y 16662874 IC50 = 101 nM T68547 CZ1OV0 16662875 IC50 = 47 nM T68547 CGQ39M 16662876 IC50 = 47 nM T68547 C5CIB4 16663079 IC50 = 59 nM T68547 CE5ZU2 16725911 IC50 > 100000 nM T68547 CUG50I 16733294 IC50 = 40.9 nM T68547 CWO7V0 16733295 IC50 = 152 nM T68547 C4W0PG 16733410 IC50 = 26.7 nM T68547 C0MO3Z 16733411 IC50 = 8.5 nM T68547 C3QL4X 16733412 IC50 = 11900 nM T68547 CV54SY 16733414 IC50 = 3220 nM T68547 C1VCX2 16733415 IC50 = 130 nM T68547 CXN07K 16733416 IC50 = 10800 nM T68547 CP9AR8 16733417 IC50 = 36.9 nM T68547 CUE62T 16733590 IC50 = 5260 nM T68547 CWUJ07 16770849 IC50 > 50000 nM T68547 CB4IN2 16773791 IC50 = 2000 nM T68547 C0ZWD2 17747368 IC50 > 10000 nM T68547 CS3PJ9 17747369 IC50 = 3700 nM T68547 CKM7F9 17747371 EC50 = 9000 nM T68547 CA5RT9 17755228 IC50 = 1200 nM T68547 CZ79PM 17756301 IC50 = 690 nM T68547 CT7K6N 17756302 IC50 = 880 nM T68547 C9MNR8 17756303 IC50 = 89 nM T68547 CU4E3H 17756304 IC50 = 410 nM T68547 CC2GS4 17756305 IC50 = 320 nM T68547 CF7JR0 17756401 IC50 = 31 nM T68547 CPVI84 17756402 IC50 = 520 nM T68547 C3FN8M 17756403 IC50 = 52 nM T68547 C5YS2I 17756404 IC50 = 200 nM T68547 C63DPZ 17756405 IC50 = 230 nM T68547 CY1V6H 17756406 IC50 = 250 nM T68547 C8GBK4 17756407 IC50 = 300 nM T68547 CZ1P9D 17756505 IC50 = 950 nM T68547 C8G9FC 17756506 IC50 = 1100 nM T68547 C5P8QU 18618646 IC50 = 1000 nM T68547 CSO6R2 20579370 IC50 = 12 nM T68547 C5S7YM 20579374 IC50 = 12 nM T68547 C09RQX 20579375 IC50 = 49 nM T68547 CXM1R3 20579392 IC50 = 12 nM T68547 CWFZ97 20579393 IC50 = 2 nM T68547 C8M6UZ 20579413 IC50 = 5 nM T68547 CQAX57 20579471 IC50 = 22 nM T68547 CU17BL 20785789 IC50 = 60 nM T68547 C9UX2V 20785858 IC50 = 200 nM T68547 CRX86F 20785861 IC50 = 100 nM T68547 CC4HZ9 20785862 IC50 = 40 nM T68547 C9TNC6 20785863 IC50 = 100 nM T68547 C1AR9N 20785977 IC50 = 22000 nM T68547 COF82Y 20785985 IC50 = 2000 nM T68547 CN4P5L 20785997 IC50 = 17000 nM T68547 CL6ZG9 20786013 IC50 = 4000 nM T68547 C4GQD8 20786025 IC50 = 17000 nM T68547 CE8O2C 20786029 IC50 = 3000 nM T68547 CPW28U 20786035 IC50 = 3000 nM T68547 CDJ6H0 20786043 IC50 = 1000 nM T68547 CES9C8 20786045 IC50 = 100 nM T68547 C7NJX8 20786052 IC50 = 300 nM T68547 CAVR26 20786058 IC50 = 300 nM T68547 CIEJ01 20786069 IC50 = 100 nM T68547 CCO6H1 20786071 IC50 = 600 nM T68547 C5ZAX8 20786082 IC50 = 100 nM T68547 C5OEY8 20786090 IC50 = 30 nM T68547 C4Q1ZB 20786113 IC50 = 100 nM T68547 CJRU62 20786114 IC50 = 30 nM T68547 CE2W3M 21630365 IC50 = 14600 nM T68547 CX91FD 22478630 IC50 = 2000 nM T68547 CLVY36 22478640 IC50 = 600 nM T68547 C5R2DE 22478644 IC50 = 4000 nM T68547 CP3OT5 22478655 IC50 = 400 nM T68547 CRZ4W0 22478660 IC50 = 100 nM T68547 C5E6CV 22478664 IC50 = 700 nM T68547 CE84LV 22478666 IC50 = 2000 nM T68547 C0PER2 22478706 IC50 = 100 nM T68547 C9VP0N 22478720 IC50 = 70 nM T68547 C13DRE 22478727 IC50 = 4000 nM T68547 CR1G5O 22478730 IC50 = 200 nM T68547 CDPF12 22478764 IC50 = 200 nM T68547 C6ME0V 22478773 IC50 = 200 nM T68547 CMY32O 22478783 IC50 = 4000 nM T68547 CI6HE2 22478790 IC50 = 300 nM T68547 CJ10DT 22478800 IC50 = 2000 nM T68547 CP2BQ1 22478822 IC50 = 80 nM T68547 C1RB5D 22478837 IC50 = 4000 nM T68547 C1CB9S 22478843 IC50 = 90 nM T68547 C9HYR1 22478847 IC50 = 200 nM T68547 CO31CW 22478851 IC50 = 200 nM T68547 CU59QK 22478870 IC50 = 2000 nM T68547 C86KRO 22478881 IC50 = 100 nM T68547 C7XJH3 22478888 IC50 = 5000 nM T68547 C6YN8U 22478891 IC50 = 3000 nM T68547 CHI9V7 22478903 EC50 = 1000 nM T68547 CAB9C4 22478932 IC50 = 3000 nM T68547 CB6QP0 22478936 IC50 = 4000 nM T68547 C7C3BW 22478949 IC50 = 3000 nM T68547 CFC28Z 22478969 IC50 = 70 nM T68547 CS5R0U 22836624 Ki = 5500 nM T68547 C2X5PQ 22958841 IC50 = 52300 nM T68547 C3CQ6Z 22986766 EC50 > 25000 nM T68547 CD2L0V 22986769 IC50 = 300 nM T68547 C1EG3M 22986772 EC50 = 5000 nM T68547 CSM54L 22986780 IC50 = 100 nM T68547 CXL02K 22986781 IC50 = 700 nM T68547 CT9M2E 22986785 IC50 = 800 nM T68547 CE3T2V 22986786 IC50 = 600 nM T68547 CKV50N 22986790 IC50 = 17000 nM T68547 C0SMZ1 23072426 IC50 = 9000 nM T68547 C9O5EB 23072489 IC50 = 6000 nM T68547 CD16PI 23521584 IC50 = 98 nM T68547 C0DFW3 23557280 IC50 = 1 nM T68547 C5E8TY 23582189 IC50 = 130 nM T68547 CEF8W4 23625604 IC50 = 3981.07 nM T68547 C5RO8F 23625605 IC50 = 1680 nM T68547 CQ12UX 23626081 IC50 = 92 nM T68547 CLM91R 23634769 IC50 = 51 nM T68547 CS58WE 23634770 IC50 = 3000 nM T68547 CF92AI 23634771 IC50 = 3800 nM T68547 CST70R 23634889 IC50 = 560 nM T68547 CX5N6D 23634890 IC50 = 1430 nM T68547 C5F9VA 23634891 IC50 = 1980 nM T68547 CE7SO1 23634892 IC50 = 1430 nM T68547 C5TH3R 23634893 IC50 = 460 nM T68547 C1WX2K 23634894 IC50 = 400 nM T68547 CN9A3R 23634895 IC50 = 2320 nM T68547 CQ6DC3 23635016 IC50 = 1030 nM T68547 CY1PR7 23635017 IC50 = 130 nM T68547 C70BKU 23640756 IC50 = 22860 nM T68547 CJYE84 23648185 IC50 = 62 nM T68547 CB8A5Q 23648260 IC50 = 190 nM T68547 C1JZ6D 23648261 IC50 = 60 nM T68547 CQJS61 23648262 IC50 = 50 nM T68547 C35ILE 23648263 IC50 = 50 nM T68547 C82BVC 23648264 IC50 > 10000 nM T68547 CT6NY2 23648265 IC50 > 10000 nM T68547 CZV0Q2 23648266 IC50 = 40 nM T68547 C36NKL 23648268 IC50 = 50 nM T68547 CS9WX8 23649315 IC50 = 250 nM T68547 CH35NV 23656767 IC50 > 100 nM T68547 CE85CP 23657268 IC50 = 17.5 nM T68547 C92WSU 23661705 IC50 = 55 nM T68547 CU01QJ 24178404 IC50 = 4 nM T68547 C1X4NQ 24707952 IC50 = 9700 nM T68547 C4UV3T 24726843 IC50 = 5700 nM T68547 CN0A5T 24744322 IC50 = 27 nM T68547 CCPE43 24744323 IC50 = 12 nM T68547 C8RC9P 24744325 IC50 = 6 nM T68547 CC5T6J 24744326 IC50 = 11 nM T68547 CP98HS 24744473 IC50 = 17 nM T68547 CCG05Q 24744793 IC50 = 9 nM T68547 CGS47I 24744797 IC50 = 14 nM T68547 C0CHJ8 24745269 IC50 = 23 nM T68547 CT2DX6 24745764 IC50 = 120 nM T68547 CMI5E4 24746277 IC50 = 8 nM T68547 CVB7J3 24746434 IC50 = 8 nM T68547 C8EYH1 24746435 IC50 = 160 nM T68547 C28AWJ 24746436 IC50 = 10 nM T68547 CSA6C8 24746437 IC50 = 8 nM T68547 CP5G1D 24759773 IC50 = 0.01 nM T68547 C17GDO 24779722 IC50 = 53.4 nM T68547 CY12VH 24825455 Ki = 88 nM T68547 CL5YW9 24825703 IC50 = 47 nM T68547 CIO7Q6 24853792 IC50 = 670 nM T68547 CBN0J5 24853793 IC50 = 27 nM T68547 CI3B6L 24857909 IC50 = 580 nM T68547 CLT5J2 24881257 IC50 = 113 nM T68547 C5GCM1 24881328 IC50 = 97.8 nM T68547 C8QVB1 24881329 IC50 = 69.2 nM T68547 CU0AM3 24881330 IC50 = 14.5 nM T68547 CQM51L 24881331 IC50 = 18 nM T68547 C4KH8F 24881332 IC50 = 52.4 nM T68547 C1KA3V 24881333 IC50 = 69.9 nM T68547 C47APB 24881402 IC50 = 18.6 nM T68547 CSN8W1 24881403 IC50 = 33.4 nM T68547 C1UQ3K 24881404 IC50 = 27.1 nM T68547 C51TMH 24881405 IC50 = 17.6 nM T68547 C9EZI7 24881406 IC50 = 14.9 nM T68547 C6P3HS 24881407 IC50 = 68.3 nM T68547 CZ3TU1 24881464 IC50 = 70.5 nM T68547 CDI49N 24881465 IC50 = 25.9 nM T68547 CQGP87 24881466 IC50 = 23.4 nM T68547 CQC8T7 24882475 IC50 = 35 nM T68547 CS1MH8 24888322 IC50 = 11000 nM T68547 CPU1Z5 24893969 IC50 = 831 nM T68547 CP29ZE 24893970 IC50 = 1220 nM T68547 CHKZ02 24894417 IC50 = 422 nM T68547 C6BNX7 24894418 IC50 = 368 nM T68547 CQ63WU 24894419 IC50 = 7510 nM T68547 C3E0SN 24894423 IC50 = 2930 nM T68547 CA56SQ 24894517 IC50 = 7120 nM T68547 CVA4J1 24894518 IC50 = 164 nM T68547 C7FV6W 24894519 IC50 = 536 nM T68547 C8R2KN 24894520 IC50 = 946 nM T68547 C2EQS1 24894522 IC50 = 1670 nM T68547 CJWI39 24894523 IC50 = 27900 nM T68547 CJ15OF 24894524 IC50 = 10400 nM T68547 CKQZ25 24894639 IC50 = 1870 nM T68547 CITS83 24894640 IC50 = 388 nM T68547 CX3QD8 24894641 IC50 = 1160 nM T68547 CC1G2E 24894642 IC50 = 980 nM T68547 CJ64TA 24894643 IC50 = 5780 nM T68547 C1PTW8 24894644 IC50 = 328 nM T68547 CKJC01 24894645 IC50 = 712 nM T68547 C6YL4C 24894776 IC50 = 2490 nM T68547 CA2O6T 24894777 IC50 = 227 nM T68547 C8XS0N 24894778 IC50 = 530 nM T68547 C6CK9N 24894779 IC50 = 1560 nM T68547 CXY5C7 24894780 IC50 = 340 nM T68547 CT4RJ0 24894895 IC50 = 587 nM T68547 CJTP74 24894896 IC50 = 762 nM T68547 C4F5TN 24894897 IC50 = 251 nM T68547 C75WEJ 24894898 IC50 = 25800 nM T68547 CMT7F4 24894899 IC50 = 592 nM T68547 CH13WV 24894900 IC50 = 672 nM T68547 CA5V7S 24894901 IC50 = 523 nM T68547 CDU08E 24895004 IC50 = 18800 nM T68547 C1IR2A 24895005 IC50 = 589 nM T68547 CQJ78L 24895006 IC50 = 3460 nM T68547 C4PN6I 24895007 IC50 = 5330 nM T68547 C9H1WI 24895008 IC50 = 501 nM T68547 CYM91Q 24895009 IC50 = 497 nM T68547 CEH9A4 24895010 IC50 = 31600 nM T68547 C8SP7C 24895115 IC50 = 887 nM T68547 C0C9VU 24895116 IC50 = 385 nM T68547 CM3Q7A 24895117 IC50 = 555 nM T68547 CZ1SP9 24895118 IC50 = 215 nM T68547 CY7D1N 24895120 IC50 = 9720 nM T68547 CH7L8Z 24895121 IC50 = 8940 nM T68547 C60FAX 24895122 IC50 = 141 nM T68547 CO68DV 24895187 IC50 = 38240 nM T68547 C40QJO 24895188 IC50 = 6110 nM T68547 C2K8BR 24895189 IC50 = 607 nM T68547 CBI25A 24895190 IC50 = 1550 nM T68547 C73LSX 24896624 IC50 = 12800 nM T68547 CC0R9O 24938735 IC50 = 0.4 nM T68547 CF03HD 24948905 IC50 = 628 nM T68547 CHP8O6 24948906 IC50 = 20.7 nM T68547 C1KRT8 24948907 IC50 = 716 nM T68547 CKY2P8 24948908 IC50 = 56.3 nM T68547 C25CFI 24948909 IC50 = 360 nM T68547 CWQ04Z 24948910 IC50 = 64.5 nM T68547 CO71ES 24950887 IC50 = 0.02 nM T68547 CM5I1O 24950892 IC50 = 0.06 nM T68547 C1JHF6 24951209 IC50 = 0.78 nM T68547 CM9I3X 24951310 IC50 = 124 nM T68547 CX1YF8 24951311 IC50 = 644 nM T68547 CV10XU 24951312 IC50 = 100 nM T68547 CD6KV0 24951313 IC50 = 826 nM T68547 CQY9Z0 24951314 IC50 = 3.2 nM T68547 C3AQG0 24957697 IC50 = 200 nM T68547 C2JZ3S 24957698 IC50 = 520 nM T68547 CZ3FO0 24958070 IC50 = 420 nM T68547 C82OXU 24958071 IC50 = 630 nM T68547 C6IC2O 24958072 IC50 = 190 nM T68547 CB16FH 24958073 IC50 = 480 nM T68547 C5H4QV 24958074 IC50 = 150 nM T68547 CCJ9G0 24958075 IC50 = 35 nM T68547 C04IDY 24958076 IC50 = 160 nM T68547 C79TOJ 24958447 IC50 = 62 nM T68547 CDTJ93 24958448 IC50 = 160 nM T68547 CSF3J5 24958449 IC50 = 130 nM T68547 CSZ1F5 24958450 IC50 = 140 nM T68547 C9QX2O 24958451 IC50 = 200 nM T68547 CAX05W 24958452 IC50 = 380 nM T68547 CH4C3E 24958809 IC50 = 150 nM T68547 CPC58S 24958810 IC50 = 120 nM T68547 C14FUP 24958811 IC50 = 390 nM T68547 CM94VS 24958812 IC50 = 350 nM T68547 C65PZU 24958813 IC50 = 420 nM T68547 C6YR5K 24958814 IC50 = 790 nM T68547 CNX41V 24958815 IC50 = 20 nM T68547 C2UZ5G 24958816 IC50 = 16 nM T68547 C8BEW0 24959168 IC50 = 78 nM T68547 CNO0U1 24959169 IC50 = 26 nM T68547 C5J3SP 24959542 IC50 = 170 nM T68547 CBM71O 24959543 IC50 = 100 nM T68547 C5BZE7 24959906 IC50 = 13 nM T68547 CC76EQ 24961017 IC50 = 41 nM T68547 CR6C3N 24962469 IC50 = 76 nM T68547 CJ1HQ5 25009146 IC50 = 230 nM T68547 C7XMO2 25009310 IC50 = 89 nM T68547 CU7G9E 25010550 IC50 = 34.67 nM T68547 CB0AY2 25012006 IC50 = 11 nM T68547 C4Q0OZ 25012007 IC50 = 9 nM T68547 CJU0D4 25012170 IC50 = 22 nM T68547 CQ94NP 25012333 IC50 = 42 nM T68547 C0EQI5 25012335 IC50 = 29 nM T68547 C5L1PC 25012495 IC50 = 21 nM T68547 C6VW2J 25012816 IC50 = 13 nM T68547 C9MCS0 25012818 IC50 = 38 nM T68547 CAJ09S 25012981 IC50 = 23 nM T68547 C5CDK0 25013299 IC50 = 20 nM T68547 CB9AD1 25013300 IC50 = 28 nM T68547 CQIW21 25013303 IC50 = 16 nM T68547 CH3KY0 25013469 IC50 = 54 nM T68547 CW31UO 25013472 IC50 = 3.5 nM T68547 CLT25N 25013473 IC50 = 7 nM T68547 CRJS45 25013632 IC50 = 6.5 nM T68547 C3UZ4M 25013789 IC50 = 140 nM T68547 CDY4R2 25013791 IC50 = 90 nM T68547 C5B0IJ 25023793 IC50 = 1400 nM T68547 CLG23N 25023794 IC50 = 12 nM T68547 CHE82I 25023795 IC50 = 7100 nM T68547 CX8G3W 25023796 IC50 = 880 nM T68547 CVRS37 25023797 IC50 = 890 nM T68547 C7GO3U 25023798 IC50 = 5000 nM T68547 C3G2AU 25023799 IC50 = 210 nM T68547 CAS18V 25023800 IC50 = 2900 nM T68547 CX7D5B 25023801 IC50 = 1300 nM T68547 CZG50I 25023802 IC50 = 4700 nM T68547 CP4T7J 25023806 IC50 = 4200 nM T68547 CF9WH6 25023808 IC50 = 9700 nM T68547 CVS1M4 25023811 IC50 = 3100 nM T68547 C9BK7U 25023852 IC50 = 138.04 nM T68547 CZP26Q 25023853 IC50 = 44.67 nM T68547 CR53MT 25023854 IC50 = 21.88 nM T68547 C0HA8S 25023855 IC50 = 27.54 nM T68547 CF67EB 25023856 IC50 = 67.61 nM T68547 C0L9PQ 25023857 IC50 = 85.11 nM T68547 CA2T1X 25023858 IC50 = 57.54 nM T68547 C7SKU1 25023859 IC50 = 30.9 nM T68547 CV8EF6 25032862 IC50 = 10 nM T68547 CX69SY 25066355 IC50 = 949 nM T68547 CF8VP4 25066356 IC50 = 560 nM T68547 CS9XH7 25066547 IC50 = 439 nM T68547 C46AGN 25066548 IC50 = 30.7 nM T68547 CJF2M7 25066549 IC50 = 204 nM T68547 CM12YX 25071720 IC50 = 92 nM T68547 CB2O3G 25072035 IC50 = 37 nM T68547 CQ5HS6 25072036 IC50 = 421 nM T68547 C9X0JM 25099146 IC50 = 960 nM T68547 CJ41EF 25099147 IC50 = 5070 nM T68547 CPTI96 25110599 IC50 = 12 nM T68547 C7ZN2W 25118059 IC50 = 1.4 nM T68547 CT08NK 25141401 IC50 = 13200 nM T68547 CGW49I 25146686 IC50 > 50000 nM T68547 C4I1CJ 25155417 IC50 = 10 nM T68547 CGU83M 25155695 IC50 = 13 nM T68547 CTK61Z 25155954 IC50 = 16 nM T68547 C72PBH 25155955 IC50 = 17 nM T68547 CB4E2J 25155956 IC50 = 7 nM T68547 CGHZ61 25156241 IC50 = 10 nM T68547 C6Q3AX 25156527 IC50 = 10 nM T68547 CF9UX7 25156797 IC50 = 20 nM T68547 CP4C5Y 25157071 IC50 = 9 nM T68547 C10UIO 25157072 IC50 = 9 nM T68547 CP9ST1 25157370 IC50 = 13 nM T68547 C7F1GA 25157660 IC50 = 11 nM T68547 CJI1B2 25157971 IC50 = 8 nM T68547 CKG24O 25157972 IC50 = 10 nM T68547 C19JIO 25157973 IC50 = 10 nM T68547 CE2TO3 25158538 IC50 = 972 nM T68547 CUA5V3 25158540 IC50 = 112 nM T68547 C1UF3Y 25159049 IC50 = 32 nM T68547 C1L9YG 25159052 IC50 = 10 nM T68547 CFS5O4 25168576 IC50 = 7600 nM T68547 C0R5OK 25168856 IC50 = 2200 nM T68547 CO14XG 25195084 IC50 = 140 nM T68547 CE5F2V 25195975 IC50 = 8 nM T68547 CB29PE 25211681 IC50 = 160 nM T68547 CM57WO 25211776 IC50 = 2150 nM T68547 CU25TK 25211878 IC50 = 460 nM T68547 C2YG9N 25216677 IC50 > 10000 nM T68547 C5CZV0 25216678 IC50 = 150 nM T68547 CB6C2A 25216810 IC50 = 850 nM T68547 CPX03T 25217055 IC50 > 10000 nM T68547 CP26WM 25217056 IC50 = 3200 nM T68547 CBDR02 25217057 IC50 = 2900 nM T68547 C9URH7 25217288 IC50 = 2400 nM T68547 C2WH9J 25217398 IC50 = 4300 nM T68547 CSM0F2 25217513 IC50 = 390 nM T68547 C1QS6M 25218542 IC50 = 348 nM T68547 CX9K4I 25218543 IC50 = 477 nM T68547 CSTH89 25218544 IC50 = 1006 nM T68547 CW51HI 25218545 IC50 = 1620 nM T68547 CNSQ31 25218546 IC50 = 24060 nM T68547 CMQ7Y8 25218547 IC50 = 13 nM T68547 C9YW5E 25218548 IC50 = 20570 nM T68547 COBV63 25218549 IC50 = 5032 nM T68547 CEY62K 25218550 IC50 = 2013 nM T68547 CBR4V1 25218551 IC50 = 5223 nM T68547 CLUQ43 25218552 IC50 = 1568 nM T68547 CDWM75 25218553 IC50 = 7964 nM T68547 C5COM1 25218554 IC50 = 33 nM T68547 CN6XA4 25218555 IC50 = 4 nM T68547 CL8K9U 25218556 IC50 = 8 nM T68547 C9WA4B 25218557 IC50 = 16 nM T68547 CRG29Y 25218558 IC50 = 47 nM T68547 CEH71M 25218560 IC50 = 11 nM T68547 CIZD97 25218561 IC50 = 11 nM T68547 C7I5EL 25218562 IC50 = 12 nM T68547 C15YDI 25218563 IC50 = 8 nM T68547 C5FZ2V 25225123 IC50 = 82600 nM T68547 CCD5M7 25227504 IC50 = 31.7 nM T68547 CK0D5S 25227505 IC50 = 78.1 nM T68547 CN97JP 25227508 IC50 = 72.2 nM T68547 CW8R1B 25227513 IC50 = 102 nM T68547 CNF50T 25229676 IC50 = 8 nM T68547 CPNQ02 25257992 IC50 = 77 nM T68547 CE0NV4 25257993 IC50 = 2.68 nM T68547 C43BHY 25269097 IC50 = 16 nM T68547 CN7K1S 25374100 IC50 = 9800 nM T68547 CU53WB 42596953 IC50 = 35 nM T68547 CJ1RQ7 42598706 IC50 = 1140 nM T68547 C2LES7 42599455 IC50 = 3.5 nM T68547 C2KO0F 42599456 IC50 = 2.9 nM T68547 C1UAO7 42601485 IC50 = 7.7 nM T68547 C3P6NY 42601488 IC50 = 200 nM T68547 COI7Y3 42611300 IC50 = 26 nM T68547 CU23PG 42611301 IC50 = 2 nM T68547 C3ZV9H 42611302 IC50 = 2700 nM T68547 CW1G2R 42611390 IC50 = 12 nM T68547 C4MP1X 42611392 IC50 = 6500 nM T68547 C62QFJ 42611486 IC50 = 30 nM T68547 CQ37HN 42612743 IC50 = 1.95 nM T68547 CX1UT9 42612744 IC50 = 544.1 nM T68547 CLH2Q7 42612852 IC50 = 116 nM T68547 CXK4C1 42618298 IC50 = 0.6 nM T68547 C7GIQ3 42625508 IC50 = 77 nM T68547 CVZ83M 42625582 IC50 = 208 nM T68547 C5MD9E 42625892 IC50 = 1160 nM T68547 CDT65Y 42631047 IC50 > 100000 nM T68547 CB79DG 42637299 IC50 > 10000 nM T68547 CP36KB 42637300 IC50 > 100000 nM T68547 CI8J6H 42637372 IC50 = 2200 nM T68547 C5RYO0 42637373 IC50 > 100000 nM T68547 CJ0CG5 42638004 IC50 > 100000 nM T68547 C8X0TG 42638005 IC50 = 2800 nM T68547 C3LHF9 42917485 IC50 = 27500 nM T68547 CO57GS 44138033 IC50 = 1820 nM T68547 C8QYH1 44157819 IC50 = 8 nM T68547 CGM5Z2 44157820 IC50 = 30 nM T68547 CQ7YU6 44157821 IC50 = 17 nM T68547 CY54FP 44157822 IC50 = 39 nM T68547 C2GPU8 44158009 IC50 = 22 nM T68547 CJR5C2 44158010 IC50 = 4 nM T68547 C0QCX7 44158079 IC50 = 2 nM T68547 C36AKC 44158080 IC50 = 51 nM T68547 C6LTW2 44158081 IC50 = 8 nM T68547 CNBD42 44158082 IC50 = 8 nM T68547 CW4IX9 44178888 IC50 = 25 nM T68547 C7RCY4 44178890 IC50 = 7 nM T68547 C4TMP9 44205087 IC50 = 3 nM T68547 CQ2VD5 44219634 IC50 = 139 nM T68547 CAG5L0 44228659 IC50 = 590 nM T68547 CMKQ59 44233027 IC50 = 3 nM T68547 CX04VN 44234773 IC50 = 1 nM T68547 C0JY2Q 44249789 IC50 = 4700 nM T68547 CU7SL0 44249820 IC50 = 9200 nM T68547 CY0QB9 44253226 IC50 = 93.8 nM T68547 C6M5XJ 44268300 EC50 = 820 nM T68547 CL80GX 44328682 IC50 = 1000 nM T68547 C12ISL 44328803 IC50 = 600 nM T68547 CCI8F7 44328901 IC50 = 4000 nM T68547 C3GRM6 44328902 IC50 = 3000 nM T68547 CW3D8V 44328913 IC50 = 1000 nM T68547 CZG57F 44328914 IC50 = 4000 nM T68547 C6RLC5 44328915 IC50 = 4000 nM T68547 C6AUY0 44328918 IC50 = 8000 nM T68547 C8R4IO 44328919 IC50 = 12000 nM T68547 C86IOC 44328927 IC50 = 740 nM T68547 C1NL0Q 44328959 IC50 = 4000 nM T68547 C9C5VS 44328965 IC50 = 3000 nM T68547 C4ER7O 44328966 IC50 = 5000 nM T68547 CC8OK4 44328974 IC50 = 4000 nM T68547 C96CLW 44328975 IC50 = 3000 nM T68547 CH7VS1 44329159 IC50 = 10000 nM T68547 CK6NG2 44329200 IC50 = 1000 nM T68547 C2O7MW 44329201 IC50 = 500 nM T68547 C42PYJ 44329220 IC50 = 5000 nM T68547 C7G5CO 44359547 IC50 = 810 nM T68547 CIT7A9 44359548 IC50 = 49000 nM T68547 CUM0Q6 44359555 IC50 = 5700 nM T68547 C2V4DN 44359681 IC50 = 1300 nM T68547 CWY06M 44363182 EC50 = 1900 nM T68547 CN91KP 44363187 EC50 = 110 nM T68547 CH4C6S 44380172 IC50 = 40 nM T68547 C1JER9 44380184 IC50 = 400 nM T68547 CP7O1B 44414162 IC50 = 10000 nM T68547 C2R7VD 44414163 IC50 = 5000 nM T68547 CKN50W 44414178 IC50 = 4000 nM T68547 C73ISD 44418011 IC50 = 3200 nM T68547 CZ1C3G 44418012 IC50 > 5000 nM T68547 CWJ51T 44418013 IC50 = 350 nM T68547 CTCJ50 44418022 IC50 = 18 nM T68547 C8KD9Z 44418025 IC50 = 25 nM T68547 CZI9M8 44418029 IC50 = 190 nM T68547 CE63RT 44418033 IC50 = 560 nM T68547 C71CHX 44418034 IC50 > 5000 nM T68547 CU35SP 44418036 IC50 > 5000 nM T68547 CBD2X6 44418037 IC50 = 930 nM T68547 CX3TJ2 44418040 IC50 = 100 nM T68547 C7FZN3 44418042 IC50 = 590 nM T68547 CE0U2L 44418046 IC50 = 33 nM T68547 CMB02F 44418058 IC50 = 180 nM T68547 CN93HS 44418061 IC50 = 480 nM T68547 CFXV51 44418062 IC50 = 3300 nM T68547 C73ELG 44418066 IC50 = 540 nM T68547 C79BSL 44418069 IC50 = 79 nM T68547 C4GP5L 44418072 IC50 = 55 nM T68547 CJ40EQ 44418074 IC50 = 44 nM T68547 CB9Q3L 44418078 IC50 = 230 nM T68547 C6GO4X 44418079 IC50 = 23 nM T68547 C0VZO8 44418083 IC50 = 200 nM T68547 C6X3TP 44418089 IC50 = 2000 nM T68547 C8MZ7R 44418110 IC50 = 22.1 nM T68547 CNV3R8 44418112 IC50 = 16 nM T68547 C5ZX0J 44418116 IC50 = 5 nM T68547 C6JD0W 44418122 IC50 = 48 nM T68547 C6OWH1 44418126 IC50 = 581 nM T68547 CY9P8C 44418127 IC50 = 80 nM T68547 C4Q3MT 44418129 IC50 = 50 nM T68547 C07ERY 44418132 IC50 = 16 nM T68547 CK3VU0 44418136 IC50 = 12.8 nM T68547 CZ74JB 44418137 IC50 = 69 nM T68547 C1PRI2 44418143 IC50 = 19 nM T68547 CJ1PU9 44418149 IC50 = 9 nM T68547 CMK6D5 44418152 IC50 = 9 nM T68547 C3KD1J 44418154 IC50 = 31 nM T68547 CP72XR 44418156 IC50 = 15.3 nM T68547 CRH1E0 44418161 IC50 = 14.3 nM T68547 C1A3TF 44418162 IC50 = 22.4 nM T68547 C41WTR 44418164 IC50 = 35 nM T68547 C5MVF9 44418166 IC50 = 34 nM T68547 C6IBO4 44418169 IC50 = 13 nM T68547 CU37ON 44418170 IC50 = 107 nM T68547 C6VC3A 44418174 IC50 = 9 nM T68547 C7D8PJ 44418178 IC50 = 8 nM T68547 CC1ZY7 44418180 IC50 = 7 nM T68547 C5Q2SD 44418181 IC50 = 8 nM T68547 C9FJ3L 44418183 IC50 = 23.5 nM T68547 CT81MK 44418184 IC50 = 8 nM T68547 CHI4U8 44418188 IC50 = 2 nM T68547 C9T8DO 44418189 IC50 = 70 nM T68547 CK26EA 44418190 IC50 = 13.1 nM T68547 CV0I5E 44418191 IC50 = 5 nM T68547 CTN6G4 44418194 IC50 = 22 nM T68547 CT2DL9 44418195 IC50 = 20 nM T68547 CY65SD 44418197 IC50 = 11 nM T68547 CME70J 44418201 IC50 = 18 nM T68547 CJAB06 44418207 IC50 = 6 nM T68547 CYJA40 44418208 IC50 = 359 nM T68547 CE10JK 44418210 IC50 = 16.4 nM T68547 CJ73PD 44418212 IC50 = 4 nM T68547 CRPD85 44418220 IC50 = 13 nM T68547 C6OB0W 44418221 IC50 = 9 nM T68547 C45BTR 44418226 IC50 = 11 nM T68547 CKXB52 44418228 IC50 = 7 nM T68547 C9R6XW 44418235 IC50 = 9 nM T68547 CFQ1G4 44418236 IC50 = 12 nM T68547 C75WVJ 44418238 IC50 = 22 nM T68547 CCAE59 44418241 IC50 = 6 nM T68547 CR45QE 44418244 IC50 = 17 nM T68547 C0OD1Z 44418245 IC50 = 8 nM T68547 CG8H9N 44418248 IC50 = 30 nM T68547 CDNR36 44418252 IC50 = 12 nM T68547 CB4ZD2 44418258 IC50 = 9 nM T68547 CY73XT 44418259 IC50 = 14 nM T68547 CE5G2H 44418267 IC50 = 8 nM T68547 C6ENC3 44427332 IC50 = 6990 nM T68547 C5YRC9 44431499 IC50 = 84000 nM T68547 CHF80J 44433619 IC50 = 963 nM T68547 CF62ER 44433620 IC50 = 168 nM T68547 C6FD8S 44433621 IC50 = 307 nM T68547 CCG3Z2 44433622 IC50 = 189 nM T68547 CMF4Q7 44433623 IC50 = 68 nM T68547 CFE3X4 44433624 IC50 = 235 nM T68547 C56OAW 44433625 IC50 = 167 nM T68547 CU2XJ7 44433626 IC50 = 39 nM T68547 C3VIF7 44433627 IC50 = 54 nM T68547 CR6ZN7 44433628 IC50 = 405 nM T68547 C2LKQ1 44433629 IC50 = 669 nM T68547 CJI1D0 44433630 IC50 = 67 nM T68547 C6IZA0 44433631 IC50 = 91 nM T68547 CE90PA 44433632 IC50 = 167 nM T68547 CF0WH3 44433633 IC50 = 82 nM T68547 CVE2A4 44433634 IC50 = 139 nM T68547 CW1YS6 44433635 IC50 = 222 nM T68547 CIAQ08 44433636 IC50 = 92 nM T68547 C4IWE2 44440542 IC50 = 11.1 nM T68547 CR5G4D 44440547 IC50 = 10 nM T68547 C09YVB 44440549 IC50 = 4 nM T68547 C2DT6L 44440559 IC50 = 1.3 nM T68547 CI9BH1 44440565 IC50 = 120 nM T68547 CX16UT 44440676 IC50 = 630 nM T68547 CDZL65 44440677 IC50 = 615 nM T68547 C9LY7W 44440678 IC50 = 600 nM T68547 CF0KX1 44440679 IC50 = 75 nM T68547 C1ZSM9 44440680 IC50 = 60 nM T68547 CFS1U9 44440681 IC50 = 155 nM T68547 CW80FD 44440682 IC50 = 285 nM T68547 C5TNQ3 44440684 IC50 = 20 nM T68547 CIY2O6 44440685 IC50 = 60 nM T68547 C9QX1E 44440687 IC50 = 45 nM T68547 CP61VX 44440688 IC50 = 175 nM T68547 CI9P5G 44440689 IC50 = 50 nM T68547 CLBK43 44440691 IC50 = 145 nM T68547 C20CBA 44440692 IC50 = 128 nM T68547 C3G8FE 44442351 IC50 = 5 nM T68547 C6YNV8 44442352 IC50 = 45 nM T68547 CFD92O 44442354 IC50 = 48 nM T68547 C1QMI0 44442356 IC50 = 94 nM T68547 C2L0CI 44442357 IC50 = 198 nM T68547 C97JRK 44442359 IC50 = 47 nM T68547 C3U8EF 44442437 IC50 = 230 nM T68547 C9ZUW5 44442438 IC50 = 220 nM T68547 CJ6SN4 44442439 IC50 = 3300 nM T68547 CP71RI 44445956 IC50 = 38 nM T68547 C3KLP5 44445957 IC50 = 38 nM T68547 CF9RX6 44445958 IC50 = 58 nM T68547 CBI5C1 44446463 IC50 = 200 nM T68547 CA0YE3 44446464 IC50 = 300 nM T68547 C6NEO3 44446465 EC50 = 2000 nM T68547 CV7P0C 44447120 IC50 = 210 nM T68547 CNC51G 44447194 IC50 = 10 nM T68547 C90YQD 44452393 IC50 = 28440 nM T68547 COW2C1 44452422 IC50 = 10300 nM T68547 CAY46N 44452443 IC50 = 6350 nM T68547 CWRM21 44452444 IC50 = 10540 nM T68547 CRP6H9 44452468 IC50 = 2980 nM T68547 CN2GF3 44452469 IC50 = 9760 nM T68547 C9FL6O 44452486 IC50 = 2610 nM T68547 C0HP2A 44452501 IC50 = 19190 nM T68547 C0HR3Q 44452526 IC50 = 3340 nM T68547 CUO4I3 44452552 IC50 = 38280 nM T68547 C78CAQ 44452557 IC50 = 16750 nM T68547 CYBU71 44452577 IC50 = 9540 nM T68547 C8WKU9 44453790 IC50 = 73 nM T68547 CHUE01 44454065 IC50 > 50000 nM T68547 CC5S0M 44454067 IC50 = 4500 nM T68547 CIOS98 44454068 IC50 > 50000 nM T68547 C0J7EA 44454069 IC50 > 50000 nM T68547 CB6YT0 44454095 IC50 = 7 nM T68547 CC8Q3T 44454096 IC50 > 50000 nM T68547 CB89WF 44454097 IC50 = 28 nM T68547 CY4L3Z 44454123 IC50 = 18 nM T68547 C5VP4D 44454144 IC50 = 48 nM T68547 CYZ3G6 44454146 IC50 > 50000 nM T68547 CQPX45 44454172 IC50 > 50000 nM T68547 CP3X8U 44454174 IC50 > 50000 nM T68547 CVJY03 44454175 IC50 > 50000 nM T68547 C8SQ2L 44454177 IC50 = 1500 nM T68547 CN9TG5 44454199 IC50 = 13000 nM T68547 C9N2QJ 44454200 IC50 > 50000 nM T68547 CIOH21 44454201 IC50 = 1300 nM T68547 C0VXC1 44454224 IC50 > 50000 nM T68547 CLRQ84 44454225 IC50 = 2100 nM T68547 CMIC06 44454226 IC50 = 250 nM T68547 C7ITR4 44454228 IC50 = 5300 nM T68547 C1RMS2 44454255 IC50 = 140 nM T68547 C7NPV1 44454256 IC50 = 330 nM T68547 C5R8LZ 44454257 IC50 > 50000 nM T68547 C6TDL4 44454282 IC50 > 50000 nM T68547 C0B3MD 44454284 IC50 > 50000 nM T68547 CNJ09C 44454348 IC50 > 50000 nM T68547 C57GMR 44454349 IC50 > 50000 nM T68547 C07UCT 44454350 IC50 > 50000 nM T68547 CX3G0B 44454376 IC50 = 44000 nM T68547 CEMP32 44454378 IC50 = 650 nM T68547 C07XZP 44454379 IC50 = 670 nM T68547 CO86JR 44454380 IC50 = 4200 nM T68547 CB1TH4 44454412 IC50 = 160 nM T68547 CGA78T 44454413 IC50 = 1000 nM T68547 C7L9EU 44454417 IC50 = 52 nM T68547 C2KF1U 44454497 IC50 = 1200 nM T68547 CH9VX0 44454499 IC50 = 610 nM T68547 C4DXH2 44454531 IC50 > 50000 nM T68547 C89PYN 44454532 IC50 = 400 nM T68547 C7GWO4 44454563 IC50 = 440 nM T68547 C86BAQ 44454564 IC50 = 1800 nM T68547 CRD24M 44454592 IC50 = 100 nM T68547 CHTW62 44454593 IC50 = 350 nM T68547 CL2SZ9 44454594 IC50 = 130 nM T68547 CO2XJ5 44454598 IC50 = 70 nM T68547 CX40AR 44454621 IC50 = 130 nM T68547 CL2H3W 44454622 IC50 = 68 nM T68547 C58DBM 44454623 IC50 = 75 nM T68547 C9WDR3 44454646 IC50 = 310 nM T68547 C56MYC 44454898 IC50 > 50000 nM T68547 C8A1ZD 44456564 IC50 = 1.8 nM T68547 CT19ZV 44456601 IC50 = 700 nM T68547 CBR4K5 44456917 IC50 = 2000 nM T68547 C9TFS1 44456918 IC50 = 3000 nM T68547 C2UE5H 44456919 EC50 = 25000 nM T68547 C5IJU1 44456955 IC50 = 159 nM T68547 CJ0L4C 44456965 IC50 = 55 nM T68547 CN9RU3 44456967 IC50 = 79 nM T68547 CO4R1Y 44456968 IC50 = 55 nM T68547 CBZU87 44456990 IC50 < 390 nM T68547 CJ31FN 44456991 IC50 = 18 nM T68547 CU03FR 44456996 IC50 = 46.5 nM T68547 C8G0PO 44457001 IC50 = 36.5 nM T68547 CM0QI2 44457003 IC50 = 26.5 nM T68547 CT32KR 44457008 IC50 = 190 nM T68547 CP73YR 44457010 IC50 = 4000 nM T68547 CI65BM 44457019 IC50 = 25 nM T68547 C8VH1E 44457028 IC50 = 3400 nM T68547 CXT7P5 44457031 IC50 = 53 nM T68547 CH72DO 44457032 IC50 = 76 nM T68547 C2TJX7 44457033 IC50 = 13 nM T68547 CWLH02 44457049 IC50 = 582 nM T68547 C74LTB 44506448 IC50 = 19 nM T68547 C2UZ1P 44507247 IC50 = 69 nM T68547 C4ME5R 44507942 IC50 > 25000 nM T68547 C92UDN 44541230 IC50 > 10000 nM T68547 C7IB2P 44541231 IC50 > 10000 nM T68547 C4TGM5 44541232 IC50 = 2500 nM T68547 CR7W5C 44541233 IC50 > 1000 nM T68547 CFXD49 44541234 IC50 > 10000 nM T68547 C4FKU6 44541235 IC50 = 3890 nM T68547 CE52NP 44543401 IC50 > 10000 nM T68547 CQI7O3 44543402 IC50 > 20000 nM T68547 CJ0KH8 44543403 IC50 > 10000 nM T68547 C7H4FD 44543404 IC50 = 2700 nM T68547 CGS14Q 44543405 IC50 = 910 nM T68547 CHX48R 44543406 IC50 > 10000 nM T68547 CG2AE4 44543407 IC50 > 1000 nM T68547 C7F8YJ 44543715 Ki = 55 nM T68547 CW4KH2 44551271 IC50 = 2000 nM T68547 C17BGM 44561972 IC50 = 24100 nM T68547 C04SOM 44561973 IC50 = 12600 nM T68547 C5RD6F 44561974 IC50 = 15700 nM T68547 CA7CG3 44561975 IC50 = 11040 nM T68547 C3UV7C 44561976 IC50 = 3770 nM T68547 C61AMY 44562034 IC50 = 4720 nM T68547 C4HQ8S 44562035 IC50 = 4290 nM T68547 C7PKX5 44562036 IC50 = 14980 nM T68547 C92FSV 44562037 IC50 = 11550 nM T68547 CX6NB4 44562038 IC50 = 49150 nM T68547 CV28HM 44562039 IC50 = 43100 nM T68547 C5CTG9 44562040 IC50 = 47070 nM T68547 CT65QO 44562076 IC50 = 29600 nM T68547 C3P0TE 44562077 IC50 = 25310 nM T68547 CCUP97 44562078 IC50 = 50140 nM T68547 CG3P8O 44562079 IC50 = 49400 nM T68547 CU92TP 44562080 IC50 = 13410 nM T68547 CW42BX 44562604 IC50 = 6800 nM T68547 CDW54Z 44562605 IC50 = 1800 nM T68547 C1WY8L 44562606 IC50 = 2900 nM T68547 C9MB4K 44562607 IC50 = 2600 nM T68547 CH2NP3 44562608 IC50 = 6540 nM T68547 CBYZ26 44562609 IC50 = 17500 nM T68547 CZU3I7 44562657 IC50 > 10000 nM T68547 C3QSI4 44562762 IC50 = 5900 nM T68547 CRJS52 44562763 IC50 = 4200 nM T68547 C2LH1N 44562764 IC50 > 5000 nM T68547 CJ5US8 44562765 IC50 = 16600 nM T68547 CUT7L8 44562766 IC50 = 2800 nM T68547 CH2KM0 44562767 IC50 = 2200 nM T68547 CQX1R2 44562798 IC50 > 10000 nM T68547 CQ5RJ3 44562799 IC50 = 990 nM T68547 C96LVR 44562800 IC50 = 5900 nM T68547 CDY0E1 44562801 IC50 = 1170 nM T68547 CEM91G 44562802 IC50 = 4800 nM T68547 CEA9D0 44562840 IC50 = 6550 nM T68547 C3DMN0 44563197 IC50 = 467 nM T68547 CGF8R5 44563236 IC50 = 7400 nM T68547 CT63QG 44563237 IC50 = 2970 nM T68547 CH43AS 44564566 IC50 > 100000 nM T68547 CIO34V 44564642 Ki = 15 nM T68547 CDE7H1 44564880 IC50 = 1100 nM T68547 CIC14U 44565181 IC50 > 10000 nM T68547 C2NYZ4 44565182 IC50 = 1300 nM T68547 CTUG48 44568433 IC50 = 725 nM T68547 CV4M2F 44570642 IC50 = 180 nM T68547 CMS4K1 44570643 IC50 = 200 nM T68547 CU69ZW 44570644 IC50 = 70 nM T68547 CJ18SD 44570805 IC50 = 170 nM T68547 CL12TK 44570806 IC50 = 50 nM T68547 C7BMS4 44570807 IC50 = 80 nM T68547 CL2F0W 44570808 IC50 = 90 nM T68547 CF5Z9M 44570853 IC50 = 160 nM T68547 CJ6T0C 44570854 IC50 = 250 nM T68547 CAR98K 44570855 IC50 = 230 nM T68547 CIRC83 44570856 IC50 = 420 nM T68547 C6HQ9U 44570890 IC50 = 250 nM T68547 CIB94L 44570891 IC50 = 190 nM T68547 CZ15BG 44570892 IC50 = 70 nM T68547 C2Y4VO 44570893 IC50 = 140 nM T68547 C4Z8YI 44570929 IC50 = 210 nM T68547 CF9U5R 44570930 IC50 = 90 nM T68547 C86XEZ 44570931 IC50 = 80 nM T68547 C0M9SB 44570973 IC50 = 140 nM T68547 CF1YN3 44570974 IC50 = 120 nM T68547 C4JC5Z 44570975 IC50 = 130 nM T68547 C2MJ1Z 44571303 IC50 > 20000 nM T68547 CN0P4C 44571304 IC50 > 20000 nM T68547 CN0WI6 44571333 IC50 = 2000 nM T68547 CRH51O 44571334 IC50 = 1200 nM T68547 CZ50XH 44571335 IC50 = 90 nM T68547 CUO3V0 44572289 IC50 = 2500 nM T68547 CFH95O 44572348 IC50 = 1500 nM T68547 CD17KA 44572349 IC50 = 4500 nM T68547 CU4VC9 44572350 IC50 = 3600 nM T68547 C5TBI9 44572351 IC50 = 350 nM T68547 COM65J 44572384 IC50 = 740 nM T68547 CV91YE 44572385 IC50 = 270 nM T68547 CAUH07 44572405 IC50 > 10000 nM T68547 CUO41X 44572406 IC50 = 120 nM T68547 CY0I4X 44572407 IC50 = 460 nM T68547 C3CB2K 44572429 IC50 = 620 nM T68547 CM2Q8J 44572430 IC50 = 230 nM T68547 CAN4B0 44572431 IC50 = 760 nM T68547 C8AO6P 44572466 IC50 = 520 nM T68547 C2O3IS 44572467 IC50 > 10000 nM T68547 CH09QJ 44572468 IC50 = 570 nM T68547 CMAT21 44572489 IC50 = 230 nM T68547 CU1SY9 44572490 IC50 = 170 nM T68547 CSD74G 44572491 IC50 = 450 nM T68547 CZ2X7L 44572516 IC50 = 700 nM T68547 CW7BK3 44572517 IC50 = 2300 nM T68547 C59TVW 44572518 IC50 = 350 nM T68547 CC74WS 44572519 IC50 = 1400 nM T68547 CA9WO3 44572537 IC50 = 310 nM T68547 C06SLW 44572538 IC50 = 470 nM T68547 CY8TG3 44572539 IC50 = 1130 nM T68547 C1JR4C 44572540 IC50 = 210 nM T68547 CV50NO 44572558 IC50 = 64 nM T68547 CB9Z4E 44572559 IC50 = 4900 nM T68547 C0RUB9 44572560 IC50 = 790 nM T68547 CY78SZ 44572561 IC50 = 500 nM T68547 CZ0PA9 44572581 IC50 = 170 nM T68547 CD9VR5 44572582 IC50 = 100 nM T68547 CG5UK0 44572584 IC50 = 160 nM T68547 CMX32U 44572633 IC50 = 120 nM T68547 CA3UR6 44572654 IC50 = 290 nM T68547 CL2M3I 44574064 IC50 = 27 nM T68547 CYW58B 44574065 IC50 = 28 nM T68547 CP0DC3 44574066 IC50 = 3 nM T68547 CK0R8J 44574067 IC50 = 34 nM T68547 C48KFZ 44574068 IC50 = 47 nM T68547 CWT0P7 44574069 IC50 = 94 nM T68547 CC5BQ4 44574070 IC50 = 120 nM T68547 CFGY42 44574099 IC50 = 23 nM T68547 C7U2RW 44574100 IC50 = 73 nM T68547 CBZV14 44574101 IC50 = 40 nM T68547 CAI7O5 44574123 IC50 = 35 nM T68547 C9HVE5 44574124 IC50 = 19 nM T68547 C24XFN 44574125 IC50 = 66 nM T68547 CN71IK 44574126 IC50 = 480 nM T68547 C09PTC 44574127 IC50 = 1000 nM T68547 C1ZKO7 44574128 IC50 = 200 nM T68547 C9E5WJ 44574129 IC50 = 170 nM T68547 CH59TE 44574130 IC50 = 350 nM T68547 C08JKG 44574131 IC50 = 110 nM T68547 CMA3R6 44574139 IC50 = 303 nM T68547 C5KLR7 44574177 IC50 > 30000 nM T68547 CFS49I 44574178 IC50 > 30000 nM T68547 CJ32DK 44574179 IC50 > 30000 nM T68547 CQOS28 44574180 IC50 = 328 nM T68547 CN96ZV 44574181 IC50 = 885 nM T68547 CWJA85 44574206 IC50 = 17100 nM T68547 C46XHW 44574207 IC50 = 12300 nM T68547 C3RY9V 44574208 IC50 = 920 nM T68547 C7DS4E 44585337 IC50 = 5130 nM T68547 C3UH5B 44589485 IC50 = 710 nM T68547 CN3J8S 44589486 IC50 = 220 nM T68547 C09TKL 44589487 IC50 = 250 nM T68547 CNO7Z1 44589488 IC50 = 500 nM T68547 CKU85Z 44589520 IC50 = 7 nM T68547 CY1AU2 44589523 IC50 = 190 nM T68547 C7GBY8 44589555 IC50 = 220 nM T68547 C9S6YH 44589556 IC50 = 100 nM T68547 CB8Z7A 44589557 IC50 = 75 nM T68547 CSHM24 44589558 IC50 = 90 nM T68547 CGP6T2 44589631 IC50 = 180 nM T68547 CNQ2E6 44589632 IC50 = 380 nM T68547 C8BG6C 44589633 IC50 = 50 nM T68547 CGI82R 44589670 IC50 = 120 nM T68547 CI93GP 44589671 IC50 = 480 nM T68547 C8GF0R 44589672 IC50 > 500 nM T68547 C1I0OQ 44589673 IC50 = 240 nM T68547 CEI5X9 44589708 IC50 = 180 nM T68547 CGE42A 44589709 IC50 > 5000 nM T68547 C14PBL 44589710 IC50 > 1500 nM T68547 CS4JP5 44589733 IC50 = 4400 nM T68547 CEPG12 44589734 IC50 = 830 nM T68547 CZVO54 44589735 IC50 = 1600 nM T68547 CPB1G7 44589736 IC50 = 1300 nM T68547 CZ7VE6 44589745 IC50 = 16 nM T68547 CDH14U 44589746 IC50 = 74 nM T68547 CN18IR 44589774 IC50 = 1600 nM T68547 CT7F0N 44589856 IC50 = 11 nM T68547 C3C6WU 44589911 IC50 = 36 nM T68547 CVA4I9 44589912 IC50 = 18 nM T68547 CVQ83W 44589913 IC50 = 22 nM T68547 CNBO74 44589970 IC50 = 8 nM T68547 C0GQ2C 44589971 IC50 = 28 nM T68547 C9OL3W 44590015 IC50 = 17 nM T68547 C5AWD8 44590016 IC50 = 6 nM T68547 C0MLS4 44590017 IC50 = 17 nM T68547 CGP0W8 44590018 IC50 = 13 nM T68547 C6F5WS 44590027 IC50 = 180 nM T68547 CD5E9Y 44590028 IC50 = 110 nM T68547 C4C5AQ 44590111 IC50 = 23 nM T68547 CGP24Y 44590116 IC50 = 270 nM T68547 CA2SJ7 44590117 IC50 = 55 nM T68547 CVPT65 44590118 IC50 = 250 nM T68547 C7VUD1 44590119 IC50 = 130 nM T68547 CVZ23T 44590151 IC50 = 13 nM T68547 CDC86A 44590152 IC50 = 29 nM T68547 CJ0U5K 44590153 IC50 = 21 nM T68547 C6VAD9 44590156 IC50 = 160 nM T68547 CF9WP7 44590157 IC50 = 300 nM T68547 CZ80UX 44590158 IC50 = 140 nM T68547 CYG7T8 44590159 IC50 = 280 nM T68547 CB67HK 44590208 IC50 = 11 nM T68547 CRG54L 44590209 IC50 = 13 nM T68547 C1G2VQ 44590210 IC50 = 16 nM T68547 CJK1Q3 44590211 IC50 = 11 nM T68547 C16-FEB 44591258 IC50 = 13 nM T68547 C3O4NM 44591285 IC50 = 490 nM T68547 CQ2WN9 44591286 IC50 > 10000 nM T68547 C8EK0X 44591287 IC50 > 10000 nM T68547 CNZ1M4 44591288 IC50 > 10000 nM T68547 C1OCI9 44591315 IC50 = 13 nM T68547 CS6P3M 44591320 IC50 > 10000 nM T68547 CJI84H 44591321 IC50 > 10000 nM T68547 CV78HA 44591322 IC50 > 10000 nM T68547 C19IEO 44591323 IC50 > 10000 nM T68547 C18NCB 44591324 IC50 > 10000 nM T68547 C82VYI 44591343 IC50 > 50000 nM T68547 CD0WI6 44592047 IC50 = 14 nM T68547 CA6Q9Y 44592060 IC50 = 6260 nM T68547 CS70EV 44592112 IC50 = 270 nM T68547 C37YMQ 44592113 IC50 = 52 nM T68547 C0AC3P 44593559 IC50 > 10000 nM T68547 CKR62F 44596100 IC50 = 3300 nM T68547 CH2J8R 44598238 IC50 = 460 nM T68547 CE5W3U 44598288 IC50 = 68 nM T68547 C68BJH 44598289 IC50 = 751 nM T68547 C9K2WV 44598290 IC50 = 136 nM T68547 C16ZEP 44598291 IC50 = 42 nM T68547 C28GHB 44598344 IC50 = 150 nM T68547 CU65LR 44598345 IC50 = 178 nM T68547 CCVA51 44598385 IC50 = 288 nM T68547 C29NXL 44598386 IC50 = 1000 nM T68547 C5WM7H 44598387 IC50 > 10000 nM T68547 CK8V9I 44598388 IC50 = 120 nM T68547 C2IS6D 44598428 IC50 = 47 nM T68547 CJ54OH 44598429 IC50 = 8 nM T68547 C3TOK2 44598431 IC50 = 56 nM T68547 CGT51H 44598480 IC50 = 20 nM T68547 CZ62IW 44598481 IC50 > 10000 nM T68547 C0OT6I 44598482 IC50 = 4840 nM T68547 CX8U6S 44598483 IC50 > 10000 nM T68547 CO5YJ8 44598535 IC50 = 200 nM T68547 C5H8RA 44598536 IC50 = 8 nM T68547 CC2QV9 44623002 IC50 > 50000 nM T68547 CVJ51M 44623152 IC50 > 50000 nM T68547 C6TJ2G 44623153 IC50 > 50000 nM T68547 CE47ZB 45102716 IC50 = 2300 nM T68547 CJWF93 45102721 IC50 = 1050 nM T68547 C42SJP 45141750 IC50 = 197 nM T68547 CLE9U5 45141751 IC50 = 200 nM T68547 COZ25S 45268021 IC50 = 532000 nM T68547 CS9DW4 45268025 IC50 = 7300 nM T68547 C0BQF9 45268900 IC50 = 191000 nM T68547 CH08UF 45268906 IC50 = 20500 nM T68547 C27VLQ 45269750 IC50 = 83900 nM T68547 CK1AP8 45269751 IC50 = 84200 nM T68547 CSM1O6 45271073 IC50 = 21000 nM T68547 C02LVF 45485792 IC50 = 8 nM T68547 C7EAV5 45485820 IC50 = 42 nM T68547 CIO0T2 46179730 IC50 = 5.06 nM T68547 C2M4GV 46179732 IC50 = 8.6 nM T68547 CS75CD 46179779 IC50 = 4.6 nM T68547 C39YKM 46179780 IC50 = 12.1 nM T68547 C0CKE5 46180624 IC50 > 30000 nM T68547 C7GYH0 46180758 IC50 = 31.9 nM T68547 C27IKH 46180759 IC50 = 8 nM T68547 CSC1Y9 46180760 IC50 = 8.7 nM T68547 C4XHL5 46180761 IC50 = 5.3 nM T68547 C70FSJ 46180763 IC50 = 5.7 nM T68547 C0W8DB 46187719 IC50 = 5170 nM T68547 CV7D4Z 46187885 IC50 = 3980 nM T68547 C53ZSX 46187886 IC50 > 10000 nM T68547 CEV52J 46187887 IC50 = 7650 nM T68547 CSC70G 46187888 IC50 > 10000 nM T68547 C7SC8A 46187889 IC50 = 8250 nM T68547 CQLG06 46187890 IC50 = 9630 nM T68547 CVGN05 46187891 IC50 > 10000 nM T68547 CF29IN 46188075 IC50 = 5320 nM T68547 COWJ59 46190552 IC50 = 5730 nM T68547 C8YO4W 46190553 IC50 = 6860 nM T68547 CEX48K 46190554 IC50 = 8320 nM T68547 C6J9DI 46190555 IC50 = 3530 nM T68547 C53RNX 46190556 IC50 > 10000 nM T68547 CPS37G 46190557 IC50 = 3850 nM T68547 C2MOT0 46190609 IC50 = 2670 nM T68547 CJ8OT2 46190610 IC50 = 9630 nM T68547 CX93ZQ 46190753 IC50 = 380 nM T68547 C85WSJ 46190754 IC50 = 2180 nM T68547 C9VEX6 46190755 IC50 = 680 nM T68547 C6O5AD 46190756 IC50 = 70 nM T68547 C7F8AM 46190820 IC50 = 1920 nM T68547 C8JY0S 46190821 IC50 = 190 nM T68547 CUCK61 46190822 IC50 = 350 nM T68547 CXQ51Y 46190823 IC50 = 490 nM T68547 CR0G9O 46190824 IC50 = 80 nM T68547 CDP80X 46190825 IC50 = 120 nM T68547 C3ETP2 46190826 IC50 = 1150 nM T68547 CZ8N7D 46197576 IC50 = 6 nM T68547 CF9QB5 46197577 IC50 = 2.8 nM T68547 CMK3H7 46197578 IC50 = 24 nM T68547 C7IGB2 46197685 IC50 = 11 nM T68547 C9T7FD 46197686 IC50 = 6 nM T68547 C8IQ5Z 46197687 IC50 = 3 nM T68547 CJZ3X6 46197795 IC50 = 16 nM T68547 C7Z6JK 46197796 IC50 = 10 nM T68547 C9Z6UF 46197797 IC50 = 19 nM T68547 CD57RJ 46197798 IC50 = 7.5 nM T68547 CR04HA 46197799 IC50 = 15 nM T68547 CFKV19 46197898 IC50 = 136 nM T68547 C3ZE2B 46198177 IC50 < 20 nM T68547 CQ83FI 46203315 IC50 = 210 nM T68547 CK8YL5 46203316 IC50 = 140 nM T68547 C1YB9P 46203618 IC50 = 910 nM T68547 C4I5DH 46203619 IC50 = 3040 nM T68547 C43KVC 46203620 IC50 = 1560 nM T68547 CY7ER9 46203621 IC50 = 4130 nM T68547 CW13ZY 46203622 IC50 = 8670 nM T68547 CND31M 46203623 IC50 = 820 nM T68547 C1RX2K 46203949 IC50 = 1050 nM T68547 CZJ86R 46203950 IC50 = 760 nM T68547 CNA07J 46203951 IC50 = 880 nM T68547 CQ69AM 46205433 IC50 = 63 nM T68547 C7V1RE 46216758 IC50 = 9.1 nM T68547 CZ0F6R 46216759 IC50 = 9.1 nM T68547 C0RQ1B 46216760 IC50 = 11 nM T68547 CI06QG 46216772 IC50 = 13 nM T68547 C5U7GY 46230638 IC50 = 25 nM T68547 CN8F9S 46830326 IC50 = 25 nM T68547 CG2R9Z 46838751 IC50 = 161.3 nM T68547 C4B7YX 46838752 IC50 = 4.5 nM T68547 C8D4XL 46861823 IC50 = 73000 nM T68547 CB2G1W 46881144 IC50 = 3.04 nM T68547 C85RDN 46881213 IC50 = 1.01 nM T68547 CQTI31 46881225 IC50 > 30000 nM T68547 C48QWG 46884058 IC50 = 1101 nM T68547 CVU0D3 46884059 IC50 = 27 nM T68547 C5UMJ3 46884060 IC50 = 149 nM T68547 CQ76JG 46884061 IC50 = 1110 nM T68547 C9HMN4 46884114 IC50 = 638 nM T68547 C8V3HK 46884115 IC50 = 1142 nM T68547 C8CI2D 46884116 IC50 = 11614 nM T68547 C35OPR 46884117 IC50 = 30 nM T68547 CI0W9C 46884118 IC50 = 17 nM T68547 CM9W8B 46886948 IC50 = 40 nM T68547 C3X1PB 46886949 IC50 = 7.9 nM T68547 CA8ZB0 46886950 IC50 = 12 nM T68547 C5STW2 46887022 IC50 = 25 nM T68547 C35ATX 46887023 IC50 = 63 nM T68547 C35LCR 46887024 IC50 = 20 nM T68547 C1C7TX 46887025 IC50 = 12 nM T68547 CC6I4F 46887026 IC50 = 12 nM T68547 CEMV64 46887060 IC50 = 10 nM T68547 CCU65S 46887061 IC50 = 16 nM T68547 C24FTM 46887062 IC50 = 10 nM T68547 C8VD6Z 46887093 IC50 = 31 nM T68547 C3UNV6 46887094 IC50 = 5 nM T68547 CJE6Q2 46887127 IC50 = 6.3 nM T68547 C4OWH7 46887128 IC50 = 5 nM T68547 C74SPT 46887178 IC50 = 10 nM T68547 C9I6NF 46887179 IC50 = 7.9 nM T68547 C28RSA 46887180 IC50 = 6.3 nM T68547 CH85NX 46887211 IC50 = 6.3 nM T68547 C8YAV5 46887212 IC50 = 10 nM T68547 CJ30VB 46887241 IC50 = 12 nM T68547 CX53HE 46887282 IC50 = 500 nM T68547 CU38FK 46887283 IC50 = 630 nM T68547 C0CTM9 46887332 IC50 = 120 nM T68547 CP4W7O 46887556 IC50 = 25 nM T68547 C2GP9T 46887557 IC50 = 63 nM T68547 C3UIY6 46887558 IC50 = 31 nM T68547 CUR2X5 46887559 IC50 = 40 nM T68547 CMU9D7 46887584 IC50 = 10 nM T68547 CA8JT1 46887585 IC50 = 16 nM T68547 C25DSY 46887918 IC50 = 67.5 nM T68547 C93CLK 46887919 IC50 = 10200 nM T68547 C5LW8V 46890006 IC50 = 43 nM T68547 C0UT9V 46890007 IC50 = 12000 nM T68547 CDZ59L 46890008 IC50 = 2420 nM T68547 C9K3FW 46890009 IC50 = 1700 nM T68547 C5KMB6 46890064 IC50 = 25 nM T68547 CL79MV 46890065 IC50 = 3750 nM T68547 C2AG8X 46890066 IC50 = 49 nM T68547 CB3LI6 46890067 IC50 = 21 nM T68547 C7UOM9 46890115 IC50 = 20 nM T68547 CL7PC8 46890116 IC50 = 34 nM T68547 C53ZYJ 46890117 IC50 = 22 nM T68547 C0QO8Y 46890540 IC50 = 245 nM T68547 CJDP81 46890581 IC50 = 115 nM T68547 C5R0PY 46890582 IC50 = 26 nM T68547 CPSI47 46890583 Ki = 8 nM T68547 CQC6A5 46890584 IC50 = 60 nM T68547 CNI41Q 46890585 IC50 = 8 nM T68547 CS57JT 46890586 IC50 = 24 nM T68547 CA4E1N 46890621 IC50 = 45 nM T68547 C5NA9Y 46890622 IC50 = 92 nM T68547 C78OFX 46890623 IC50 = 185 nM T68547 C0Y6DW 46890624 IC50 = 6 nM T68547 C6U7NG 46890625 IC50 = 44 nM T68547 C5OS8T 46890668 IC50 = 97 nM T68547 CLP8Y6 46890669 IC50 = 26 nM T68547 C3U6WX 46890670 IC50 = 1250 nM T68547 CR9K3U 46890671 IC50 = 20 nM T68547 CV0M4A 46890672 IC50 = 46 nM T68547 C90NYX 46896338 IC50 = 60 nM T68547 CJ0PA2 46906644 IC50 > 100000 nM T68547 CJZ7U3 46906689 IC50 > 100000 nM T68547 C05TZR 46906690 IC50 = 18000 nM T68547 C1DUG9 46906691 IC50 = 19000 nM T68547 CTS93V 46906692 IC50 = 1000 nM T68547 CHD3F6 46906693 IC50 = 1100 nM T68547 CQ3MO8 46906748 IC50 = 3300 nM T68547 C4B6MZ 46906749 IC50 = 900 nM T68547 CV9WE5 46906750 IC50 > 10000 nM T68547 CIO0J5 46906818 IC50 = 1200 nM T68547 C43EAQ 46906819 IC50 = 800 nM T68547 C6AH1I 46906820 IC50 = 800 nM T68547 CYUP09 46906821 IC50 = 700 nM T68547 C1HV6U 46907409 IC50 = 60 nM T68547 CXH64A 46918825 IC50 = 3162.28 nM T68547 C6GY9I 46934544 IC50 = 4950 nM T68547 C3OD2Y 46934546 IC50 = 17700 nM T68547 CI8ZX5 49799582 IC50 = 13.7 nM T68547 CL7PS1 49831258 IC50 = 45000 nM T68547 CI5L2P 49846123 IC50 = 153.91 nM T68547 C4DL0M 49847150 IC50 = 19.4 nM T68547 CC7Y9U 49850262 IC50 = 144 nM T68547 C50PXU 49855444 IC50 > 50000 nM T68547 CE7D2J 49855568 IC50 = 610 nM T68547 CFD9P3 49855569 IC50 = 24000 nM T68547 C1AU5N 49855758 IC50 = 650 nM T68547 CIFK93 49855759 IC50 > 50000 nM T68547 CK48OJ 49855760 IC50 > 50000 nM T68547 CZI3M1 49855761 IC50 > 100000 nM T68547 CRPZ58 49855949 IC50 > 100000 nM T68547 CTU0K3 49855950 IC50 > 100000 nM T68547 CF85NL 49855951 IC50 > 32000 nM T68547 CF7YS9 49855952 IC50 > 50000 nM T68547 CJU38G 49855953 IC50 = 940 nM T68547 C6POK9 49856931 IC50 = 6 nM T68547 CWP27Q 49861283 IC50 = 140 nM T68547 CUFA67 50898589 IC50 = 427 nM T68547 CPOL89 50898669 IC50 = 5190 nM T68547 CRHI06 50898670 IC50 = 4640 nM T68547 C5HPL0 50898672 IC50 = 5820 nM T68547 CC1D9T 50898753 IC50 = 8620 nM T68547 CC8F0Y 50898754 IC50 = 16400 nM T68547 CZT96S 50898755 IC50 = 2740 nM T68547 C6UOH5 50898756 IC50 = 1610 nM T68547 CB75JS 50898757 IC50 = 10200 nM T68547 C9A7XU 50898841 IC50 = 3980 nM T68547 CQ43IF 50898842 IC50 = 15700 nM T68547 CF0TI2 50898843 IC50 = 7450 nM T68547 CJ1YC2 50898949 IC50 = 10300 nM T68547 CKD7X9 50898950 IC50 = 4050 nM T68547 C9BYZ1 50899047 IC50 = 2070 nM T68547 CB89VJ 50899050 IC50 = 4320 nM T68547 C59RDT 50899051 IC50 = 9700 nM T68547 C52ABG 50942502 IC50 = 60 nM T68547 CPQ0F7 50991199 IC50 = 25 nM T68547 CSC3P9 50992051 IC50 = 7 nM T68547 CV3X4J 51033161 IC50 > 50000 nM T68547 C5LZ4R 51351536 IC50 > 30000 nM T68547 CI68XL 52912223 IC50 > 100000 nM T68547 CVLE09 52950031 IC50 > 10000 nM T68547 CE43FC 53249967 IC50 > 30000 nM T68547 C8SUQ5 53317424 IC50 > 30000 nM T68547 C7MO2J 53325871 IC50 = 3.8 nM T68547 CG84JS 53325976 IC50 = 200 nM T68547 CVM4Q3 53357987 IC50 = 1700 nM T68547 C3B5AJ 53361011 IC50 = 4 nM T68547 C78GKN 53361474 IC50 = 99.1 nM T68547 CNB63X 53361475 IC50 = 82.2 nM T68547 CS2P3T 53363085 IC50 = 53 nM T68547 COG5K0 53363092 IC50 = 1 nM T68547 CCZW39 53363093 IC50 = 3 nM T68547 C8GKN4 53363517 IC50 = 2490 nM T68547 CQ43VH 53363518 Ki = 7.7 nM T68547 C7Z6BW 53363708 IC50 = 575 nM T68547 CUY8V2 53363709 IC50 = 169 nM T68547 CZ2EP4 53363796 IC50 = 175 nM T68547 CX72IP 53363797 IC50 = 84 nM T68547 CU7VZ1 53363805 IC50 = 13 nM T68547 CN5RK6 53363806 IC50 = 120 nM T68547 CU72IM 53363807 IC50 = 210 nM T68547 CEA9B3 53363887 IC50 = 130 nM T68547 CK0R3L 53363888 IC50 = 47 nM T68547 CN27BZ 53363889 IC50 = 23 nM T68547 C4D9RH 53363970 IC50 = 1.3 nM T68547 C6N8KX 53363971 IC50 = 17 nM T68547 C1YE6I 53364276 IC50 = 11 nM T68547 CZ62DW 53364278 IC50 = 8 nM T68547 CT14SP 53364279 IC50 = 21 nM T68547 C3WBV5 53364352 IC50 = 1.5 nM T68547 CC64OS 53364353 IC50 = 10 nM T68547 CFHR93 53364354 IC50 = 6 nM T68547 C81EPA 53364355 IC50 = 6 nM T68547 CSV85J 53364356 IC50 = 2 nM T68547 C2PHM7 53364357 IC50 = 1 nM T68547 C6Y2EV 53374826 IC50 = 4110 nM T68547 CC5K2U 53380601 IC50 = 730 nM T68547 CN17BX 53380699 IC50 = 1610 nM T68547 C6X5SA 53389591 IC50 = 450 nM T68547 C9U7GF 53464577 IC50 = 12.3 nM T68547 C4EYP7 53464578 IC50 = 124.8 nM T68547 C0WNH9 53464579 IC50 = 33.2 nM T68547 C4MQ3U 53464638 IC50 = 18.1 nM T68547 CJ53ZV 53464639 IC50 = 71.2 nM T68547 CN9RH2 53464770 IC50 = 69.9 nM T68547 C0ZK7I 54576529 IC50 = 41.46 nM T68547 CTP2S1 54576530 IC50 = 42.92 nM T68547 CS8HY5 54576744 IC50 = 32.27 nM T68547 C5A7MU 54613496 IC50 = 20.2 nM T68547 CVP16C 54753629 IC50 = 22000 nM T68547 CQ1EX7 54770442 IC50 = 52.73 nM T68547 CJ1G6K 56591671 IC50 = 50 nM T68547 C7OJ4K 56602459 IC50 = 0.28 nM T68547 CT8JE7 56602463 IC50 = 0.93 nM T68547 CNJ38L 56658047 IC50 = 8 nM T68547 C1B5CM 56658048 IC50 = 8 nM T68547 CU50ZM 56658165 IC50 = 11 nM T68547 CIO96M 56659403 IC50 > 100000 nM T68547 CMW5G1 56659902 IC50 = 980 nM T68547 CT4ZY0 56661203 IC50 = 20 nM T68547 CR37GB 56661557 IC50 = 17 nM T68547 C7R9TZ 56663191 IC50 = 0.4 nM T68547 CICE56 56664976 IC50 = 9 nM T68547 CT3U2D 56665362 IC50 = 31 nM T68547 CL18NI 56666337 IC50 > 100000 nM T68547 CB3DK0 56666803 IC50 = 750 nM T68547 C07SHF 56668409 IC50 = 10 nM T68547 CQD4K8 56671918 IC50 = 9 nM T68547 CAKO50 56671919 IC50 = 14 nM T68547 CQB8V9 56671920 IC50 = 9 nM T68547 CL7SK1 56671921 IC50 = 16 nM T68547 C9LC5Y 56673234 IC50 > 100000 nM T68547 CWH5N4 56673261 IC50 > 100000 nM T68547 C1E4CX 56673467 IC50 = 130 nM T68547 CHD3I9 56673754 IC50 = 980 nM T68547 C6H3WB 56673771 IC50 = 680 nM T68547 C9YZF1 56675295 IC50 = 6 nM T68547 CFXM17 56675296 IC50 = 10 nM T68547 C0ZJG3 56676500 IC50 = 1.2 nM T68547 CG79ZX 56677183 IC50 = 32 nM T68547 CSFW85 56678631 IC50 = 6 nM T68547 C19FUS 56678632 IC50 = 10 nM T68547 CS72XM 56678633 IC50 = 15 nM T68547 C6NFB4 56678634 IC50 = 7 nM T68547 C0SN9U 56678766 IC50 = 13 nM T68547 CGCA84 56680098 IC50 = 92 nM T68547 CO69SH 56681958 IC50 = 11 nM T68547 CJ69QE 56681959 IC50 = 8 nM T68547 CMT49S 56682075 IC50 = 7 nM T68547 CR0E4M 56683440 IC50 = 89 nM T68547 C7YL4Z 56683727 IC50 = 450 nM T68547 C2ML5S 56837168 IC50 = 9.37 nM T68547 CCW89V 56932477 IC50 = 0.00687 nM T68547 C7ABK4 56933019 IC50 = 9960 nM T68547 CZ25SN 56935695 IC50 > 30000 nM T68547 CVHR15 56950025 IC50 = 22100 nM T68547 CH7W3C 56950026 IC50 = 14100 nM T68547 CLV69W 56950027 IC50 = 1880 nM T68547 C05BNS 56950152 IC50 = 1020 nM T68547 CV2X3N 56950154 IC50 = 10300 nM T68547 C83UDV 56964457 IC50 = 47 nM T68547 C3LSF8 57325671 IC50 = 4600 nM T68547 CAW53S 57325672 IC50 = 54 nM T68547 C9P8HJ 57325755 IC50 = 11 nM T68547 C6PU3K 57326321 IC50 = 11000 nM T68547 C8XVR0 57326322 IC50 = 380 nM T68547 CJY09O 57326509 IC50 = 7300 nM T68547 CS0PH3 57326510 IC50 > 50000 nM T68547 CQN86X 57326511 IC50 = 5000 nM T68547 CT58WK 57326610 IC50 = 9000 nM T68547 CP5EU9 57326611 IC50 = 50000 nM T68547 CG7S8T 57326612 IC50 = 12600 nM T68547 C7UY5V 57326613 IC50 = 6100 nM T68547 CDTL85 57326614 IC50 = 3000 nM T68547 CY0XG3 57326709 IC50 = 400 nM T68547 CG6Z2X 57326710 IC50 = 5 nM T68547 C9V5KT 57326712 IC50 = 1100 nM T68547 C4ME8Z 57326713 IC50 = 6 nM T68547 C3Y5LI 57326714 IC50 = 27 nM T68547 C5YQ3I 57326715 IC50 = 15 nM T68547 CP4EL2 57328394 IC50 = 5700 nM T68547 CO1HZ7 57331970 IC50 = 48000 nM T68547 C8EX9I 57332105 IC50 = 74000 nM T68547 CE78IS 57332106 IC50 = 57000 nM T68547 C10DMC 57336560 Ki = 7000 nM T68547 C8FLE6 57382288 IC50 = 2123 nM T68547 CW02FD 57393108 IC50 = 60 nM T68547 CX0I2Z 57396604 IC50 = 100 nM T68547 CB8N4P 57400091 IC50 = 80 nM T68547 C4LI0D 57521296 IC50 = 17000 nM T68547 C8CQ7V 57523845 IC50 = 8880 nM T68547 C4SK5V 57524018 IC50 > 100000 nM T68547 CFHU47 57524021 IC50 = 11200 nM T68547 CBZX29 57524107 IC50 = 6020 nM T68547 C5LBS0 57524273 IC50 = 19200 nM T68547 CVU30I 57524661 IC50 > 100000 nM T68547 CBM30D 57524665 IC50 = 21800 nM T68547 C3VU1R 57524666 IC50 = 12100 nM T68547 C3ZE4W 57524748 IC50 = 14300 nM T68547 CJ68EZ 57524753 IC50 = 26700 nM T68547 C4YNT9 57524833 IC50 = 17100 nM T68547 C6A3CR 57524835 IC50 = 12800 nM T68547 CTA82N 57524908 IC50 = 15900 nM T68547 CXFJ46 57550498 IC50 = 1100 nM T68547 CWT6O0 57723146 IC50 = 26 nM T68547 CA5Q6O 58147189 IC50 > 50000 nM T68547 C4DYC0 58147224 IC50 > 50000 nM T68547 CMP04X 58147302 IC50 > 50000 nM T68547 C4V7FY 58191950 IC50 = 91 nM T68547 CPCA29 58191961 IC50 = 6.5 nM T68547 C7HF1L 58191965 IC50 = 41 nM T68547 CR4BX0 58191982 IC50 = 310 nM T68547 C8V1NK 58191988 IC50 = 8600 nM T68547 C8LWY9 58191997 IC50 = 74 nM T68547 C3IQ9B 58191999 IC50 = 2200 nM T68547 CQB69R 58192003 IC50 = 10500 nM T68547 CLD40J 58465708 IC50 = 15000 nM T68547 CV9C6R 58930542 IC50 = 108 nM T68547 CI9SQ8 59033885 IC50 = 12.1 nM T68547 C1MB4Q 59323957 IC50 > 30000 nM T68547 CK6LX0 59454220 IC50 = 100 nM T68547 C2SDN1 59454252 IC50 = 140 nM T68547 CO6A2S 59585196 IC50 = 43000 nM T68547 CLN20W 60143424 IC50 = 64.7 nM T68547 CEF0C3 60143425 IC50 = 59.2 nM T68547 CRNZ07 60145504 IC50 = 65.2 nM T68547 C31TUG 60145641 IC50 = 66.9 nM T68547 CG6M7H 60145642 IC50 = 5.1 nM T68547 C8XKG0 60145643 IC50 = 71.2 nM T68547 CC72HW 60145644 IC50 = 70.9 nM T68547 CBHR24 60145645 IC50 = 64.1 nM T68547 CS85AJ 60145783 IC50 = 68.2 nM T68547 C8SZ7X 60145784 IC50 = 7.6 nM T68547 CIP62A 60145785 IC50 = 64.4 nM T68547 CZPN39 60145786 IC50 = 66.7 nM T68547 CGX45C 60145787 IC50 = 65.2 nM T68547 CPZ5Q3 60148646 IC50 > 50000 nM T68547 C8ZL3J 60148690 IC50 = 24000 nM T68547 CK5N4E 60148693 IC50 = 32000 nM T68547 C27DKW 60148711 IC50 = 21000 nM T68547 CKQ5T4 60150860 IC50 = 269 nM T68547 CS9W8Y 60151000 IC50 = 1220 nM T68547 C3TOE5 60151001 IC50 = 649 nM T68547 CR7M6T 60151002 IC50 = 252 nM T68547 CX24YF 60151004 IC50 = 107 nM T68547 C0M5BQ 60151005 IC50 = 2570 nM T68547 CDK13Q 60151006 IC50 = 202 nM T68547 C43ZUI 60151007 IC50 = 1900 nM T68547 CJ72TS 60151139 IC50 = 122 nM T68547 C5FIE4 60151140 IC50 = 3580 nM T68547 C76ENL 60151141 IC50 = 1360 nM T68547 C6KNM8 60151142 IC50 = 1680 nM T68547 CHE0N8 60151143 IC50 = 2210 nM T68547 CB35GW 60151144 IC50 = 396 nM T68547 C8H6JK 60151145 IC50 = 1050 nM T68547 C52SGF 60151146 IC50 = 807 nM T68547 CB7X2E 60151224 IC50 = 2.78 nM T68547 CY05OU 60151225 IC50 = 21.6 nM T68547 CF31LX 60151274 IC50 = 862 nM T68547 CO93CG 60151276 IC50 = 159 nM T68547 CWO8H0 60152596 IC50 = 158 nM T68547 CXW14A 60164619 IC50 = 2511.89 nM T68547 C8U2FY 60166911 IC50 = 9200 nM T68547 CVX2B7 60166912 IC50 = 1700 nM T68547 C1VQ2S 60167040 IC50 = 2900 nM T68547 C6QK1B 60167041 IC50 = 1800 nM T68547 CBOP30 60167042 IC50 = 1400 nM T68547 C97TQL 60167043 IC50 = 3100 nM T68547 CF5AE7 60167044 IC50 = 2300 nM T68547 CPF82Q 60167045 IC50 = 900 nM T68547 CNK79E 60167046 IC50 = 3600 nM T68547 C29UHY 60167191 IC50 = 7500 nM T68547 CB84PT 60167193 IC50 = 7400 nM T68547 C95XVC 60167194 IC50 = 1600 nM T68547 CS75YW 60167195 IC50 = 2900 nM T68547 C70DSE 60167196 IC50 = 2500 nM T68547 CJ6WO4 60167197 IC50 = 1000 nM T68547 C4V8TM 60167340 IC50 = 2000 nM T68547 CL4NM5 60167341 IC50 = 1400 nM T68547 CV80FM 60167342 IC50 = 700 nM T68547 CUS36O 60167343 IC50 = 3100 nM T68547 C6GIA1 60167344 IC50 = 4500 nM T68547 CQ1U0P 60200243 IC50 > 50000 nM T68547 C5F0OQ 62706003 IC50 = 140 nM T68547 CQAM69 62706004 IC50 = 70 nM T68547 C6CK5L 62706005 IC50 = 1400 nM T68547 C08BWT 62706006 IC50 = 13000 nM T68547 COTB68 62706167 IC50 = 2700 nM T68547 CM0LI9 62706168 IC50 = 3800 nM T68547 C5I8OL 62706169 IC50 = 55000 nM T68547 CW48QK 62706170 IC50 = 3800 nM T68547 CIQ52T 62706171 IC50 = 990 nM T68547 C8V2NC 62706321 IC50 = 1210 nM T68547 CUJH49 69382972 IC50 = 320 nM T68547 CBN3L0 69950064 Ki > 23000 nM T68547 C6RFQ8 70676597 IC50 = 3000 nM T68547 C5ART0 70681693 IC50 = 8900 nM T68547 CM4XB8 70681905 IC50 = 5670 nM T68547 CW5MP0 70681906 IC50 = 6080 nM T68547 CGYX13 70681907 IC50 = 6800 nM T68547 CPMZ01 70681908 IC50 = 11490 nM T68547 CD0YC8 70681968 IC50 = 2830 nM T68547 CM62BN 70682297 Ki = 49 nM T68547 C3PR4C 70684025 IC50 = 35070 nM T68547 C8R9XE 70684026 IC50 = 6800 nM T68547 CH2OA7 70684090 IC50 = 2980 nM T68547 C60XID 70684091 IC50 = 920 nM T68547 CT64UC 70686159 IC50 = 22500 nM T68547 C94YFZ 70686160 IC50 = 40120 nM T68547 C8L6YP 70686231 IC50 = 460 nM T68547 CGJK81 70686232 IC50 = 1020 nM T68547 CBZ8W0 70688300 IC50 = 39430 nM T68547 CWF4E8 70688346 IC50 = 3330 nM T68547 C31DBR 70690110 IC50 = 8600 nM T68547 C0CQP5 70690303 IC50 = 10320 nM T68547 C8T1FV 70690304 IC50 = 2960 nM T68547 CTE30H 70690378 IC50 = 3430 nM T68547 C73FOZ 70691182 IC50 > 250000 nM T68547 CQ1R3N 70692543 IC50 = 420 nM T68547 C7VF1B 70692849 Ki = 49 nM T68547 CZ0XO8 70693288 IC50 = 84000 nM T68547 CGSM24 70694519 IC50 = 2590 nM T68547 C1JO8E 70694590 IC50 = 1760 nM T68547 CWJ39I 70694591 IC50 = 1090 nM T68547 C49EGA 70694593 IC50 > 50000 nM T68547 C4W5OF 70695382 IC50 = 38000 nM T68547 CE67KO 70695508 IC50 = 6300 nM T68547 CX23AC 70696578 IC50 = 9700 nM T68547 CW6F1J 70696579 IC50 = 65710 nM T68547 C3DW5T 70696631 IC50 = 1050 nM T68547 CD5O7B 70696632 IC50 = 420 nM T68547 CEY8V3 70697398 IC50 = 80000 nM T68547 CRZ34W 70697399 IC50 = 39400 nM T68547 CQY1I6 70789579 Ki = 11900 nM T68547 C0I6VW 71139142 IC50 < 20 nM T68547 C2ED7S 71139195 IC50 < 20 nM T68547 C4BWT1 71142064 IC50 < 20 nM T68547 C8JK7A 71142076 IC50 < 20 nM T68547 C50RGP 71142078 IC50 < 20 nM T68547 CS1K8D 71142081 IC50 < 20 nM T68547 CK6GL1 71142097 IC50 < 20 nM T68547 C2RI8V 71142100 IC50 < 20 nM T68547 C6L0JF 71142106 IC50 < 20 nM T68547 C2I9UX 71142126 IC50 < 20 nM T68547 C25CUJ 71142127 IC50 < 20 nM T68547 C8NZA0 71449818 IC50 = 111000 nM T68547 C63AHI 71449819 IC50 = 86000 nM T68547 CCZ73P 71450111 IC50 = 265 nM T68547 CH2PV4 71450133 IC50 = 5180 nM T68547 C37HBI 71451928 IC50 = 8950 nM T68547 C4ZNG6 71451952 IC50 = 2250 nM T68547 C0ES2V 71453199 IC50 = 150 nM T68547 C3J9QZ 71453454 IC50 = 700 nM T68547 C9NWA2 71453740 IC50 = 1360 nM T68547 CQ1G6B 71453741 IC50 = 2550 nM T68547 CEY13X 71453772 IC50 = 1690 nM T68547 C57ATO 71455172 IC50 = 540 nM T68547 C6B2HJ 71456958 IC50 = 180 nM T68547 C57LCN 71457287 IC50 = 3120 nM T68547 C76SGF 71457594 IC50 = 990 nM T68547 C6C4OT 71458560 IC50 = 10 nM T68547 C0KRN9 71458561 IC50 = 0.4 nM T68547 CM9A3I 71458827 IC50 = 200 nM T68547 C2HZ7Q 71460412 IC50 = 190 nM T68547 CEXJ68 71460922 IC50 = 1360 nM T68547 CBK53U 71462097 IC50 = 4200 nM T68547 CXSN25 71462624 IC50 = 8120 nM T68547 CES2C4 71462625 IC50 = 1910 nM T68547 C72DJO 71465631 IC50 = 29 nM T68547 CQ7VL0 71467493 IC50 = 90 nM T68547 C5BR1D 71467494 IC50 = 120 nM T68547 CS74UB 71467495 IC50 = 1900 nM T68547 CX3U9M 71467628 IC50 = 2600 nM T68547 C3PIK2 71467958 IC50 = 210 nM T68547 CTNS49 71467959 IC50 = 610 nM T68547 CQ6B2I 71467960 IC50 = 30 nM T68547 C0YXF2 71467961 IC50 = 340 nM T68547 C1MH5Z 71467962 IC50 = 50 nM T68547 C7ESZ2 71467963 IC50 = 30 nM T68547 C45FCJ 71468055 IC50 = 120 nM T68547 C3H0CR 71468158 IC50 = 10 nM T68547 CQ26IW 71468159 IC50 = 20 nM T68547 C6ZPJ4 71468160 IC50 = 1570 nM T68547 CJU64Z 71468161 IC50 = 70 nM T68547 CD8O7W 71468162 IC50 = 350 nM T68547 CSDO79 71468163 IC50 = 630 nM T68547 CN97RG 71468164 IC50 = 110 nM T68547 C5I0TX 71468273 IC50 = 200 nM T68547 CJKU04 71468274 IC50 = 160 nM T68547 CZJ84E 71468275 IC50 = 490 nM T68547 C6L0RV 71468277 IC50 = 110 nM T68547 CAH65F 71468278 IC50 = 60 nM T68547 CVP26X 71468393 IC50 = 50 nM T68547 CFW2I5 71468672 IC50 = 23.74 nM T68547 CIS73X 71468801 IC50 = 2590 nM T68547 CS86BK 71468803 IC50 = 9690 nM T68547 CJD46S 71468805 IC50 = 2660 nM T68547 CU9FQ3 71468924 IC50 = 2450 nM T68547 C01IKD 71468927 IC50 = 450 nM T68547 CNXK19 71468928 IC50 = 240 nM T68547 C0CX7P 71476624 Ki > 2500 nM T68547 C6QPH1 71476625 Ki > 2500 nM T68547 C3JLD4 71476626 Ki > 2500 nM T68547 C3OH6T 71476627 Ki > 2500 nM T68547 C7GY8U 71495390 IC50 = 207 nM T68547 CBE46I 71495482 IC50 = 45 nM T68547 CQ5FC3 71495575 IC50 = 145 nM T68547 CIQ3E7 71495576 IC50 = 72 nM T68547 CAL79Y 71495577 IC50 = 29 nM T68547 C1SXH7 71495578 IC50 = 11 nM T68547 C1Q8LP 71495673 IC50 = 39 nM T68547 CF72JS 71495674 IC50 = 175 nM T68547 C3T7UP 71495675 IC50 = 87 nM T68547 CIW1O0 71518383 IC50 = 53 nM T68547 CY84ZI 71518384 IC50 = 35 nM T68547 C4ARY7 71518385 IC50 = 110 nM T68547 CWR36P 71518541 IC50 = 127 nM T68547 CY1KB0 71518542 IC50 = 97 nM T68547 C62ENM 71518543 IC50 = 131 nM T68547 C60KSQ 71518544 IC50 = 154 nM T68547 CU9CL6 71518545 IC50 = 97 nM T68547 CLV12J 71518706 IC50 = 135 nM T68547 CXZ0G7 71518707 IC50 = 125 nM T68547 CFQ2N9 71520536 IC50 = 189 nM T68547 C0LWJ6 71520631 IC50 = 341 nM T68547 CO28HI 71520716 IC50 = 320 nM T68547 CVA5Q7 71520717 IC50 = 320 nM T68547 C89SWX 71527724 IC50 > 30000 nM T68547 C6S5JQ 71527847 IC50 = 180.4 nM T68547 C6KBD4 71534512 IC50 = 74 nM T68547 CT51EW 71534810 IC50 = 8 nM T68547 C7QN3O 71534812 IC50 = 2 nM T68547 C8M3HU 71537640 IC50 = 53 nM T68547 C2QML7 71537641 IC50 = 7 nM T68547 CZJX53 71537927 IC50 = 2900 nM T68547 CU0ZE6 71537928 IC50 = 13 nM T68547 CH9FS7 71537929 IC50 = 92 nM T68547 CTW95A 71537931 IC50 = 12 nM T68547 C3C0RO 71538475 IC50 = 11 nM T68547 CIA28E 71538746 IC50 = 15 nM T68547 CFCV26 71538748 IC50 = 504 nM T68547 CY2T1Q 71538749 IC50 = 386 nM T68547 C4A6VJ 71538750 IC50 = 8 nM T68547 CG72NC 71538751 IC50 = 32 nM T68547 C7RUE6 71540743 IC50 = 17600 nM T68547 C9LA4F 71540744 IC50 = 2350 nM T68547 C0EK5J 71540745 IC50 = 7420 nM T68547 C80HZX 71540746 IC50 = 100 nM T68547 C4G5US 71540862 IC50 = 1670 nM T68547 C0KPM7 71542507 IC50 = 0.75 nM T68547 CX6I3N 71577043 IC50 = 6600 nM T68547 CKR6U8 71583101 IC50 = 21000 nM T68547 CBZ5S9 71583103 IC50 = 11000 nM T68547 C3PSJ9 71583105 IC50 = 12000 nM T68547 C21GHR 71624738 IC50 = 630 nM T68547 CLW8K3 71625224 IC50 = 129 nM T68547 C53BQN 71625225 IC50 = 50 nM T68547 CCQ0U1 71625341 IC50 = 369 nM T68547 COZX76 71625342 IC50 = 116 nM T68547 CD09SV 71625344 IC50 = 37 nM T68547 CM7T9N 71625573 IC50 = 1600 nM T68547 CJ6OC7 71625574 IC50 = 1850 nM T68547 CZY38J 71625575 IC50 = 601 nM T68547 C5U8OT 71625576 IC50 = 440 nM T68547 CPW9D3 71625687 IC50 = 440 nM T68547 CO62IW 71625688 IC50 = 645 nM T68547 CFP45T 71625689 IC50 = 701 nM T68547 CW1RS8 71625690 IC50 = 112 nM T68547 CXS94U 71625691 IC50 = 246 nM T68547 CU65GH 71655059 IC50 = 122 nM T68547 CPS58L 71655136 IC50 = 64.8 nM T68547 CFW7Q9 71655137 IC50 = 63.4 nM T68547 C9S0UB 71655138 IC50 = 122.9 nM T68547 CU27EV 71655139 IC50 = 125.2 nM T68547 CO8R1Z 71655216 IC50 = 159 nM T68547 C0W6EK 71655283 IC50 = 124.7 nM T68547 C7HG0K 71655802 IC50 = 638 nM T68547 CV73YD 71660259 IC50 = 1330 nM T68547 CQ5UR0 71660260 IC50 = 9580 nM T68547 CQ5P0T 71660261 IC50 = 720 nM T68547 C8EIX0 71660262 IC50 = 1600 nM T68547 CPJ4V7 71680913 IC50 = 12000 nM T68547 C3KO9V 71680916 IC50 = 39100 nM T68547 CI9G3B 71681069 IC50 = 6100 nM T68547 C5WZV9 71720123 IC50 < 20 nM T68547 CIR56T 71721558 IC50 > 100000 nM T68547 CCD18W 71721946 IC50 = 1110 nM T68547 CFUC24 71722010 IC50 = 11.1 nM T68547 CEG67K 71723449 IC50 = 490 nM T68547 CXMZ49 71732116 IC50 = 6130 nM T68547 C0H9PY 71732117 IC50 = 7540 nM T68547 CSI0W8 71732119 IC50 = 2740 nM T68547 CWGF27 71732120 IC50 = 14400 nM T68547 C0P8CH 71748076 IC50 = 4850 nM T68547 CU4X2F 71761851 IC50 = 15 nM T68547 C7SK3L 71761852 IC50 = 15 nM T68547 CI2NH1 71761853 IC50 = 75 nM T68547 CORB04 71762088 IC50 = 28 nM T68547 CYG6O7 71762089 IC50 = 28 nM T68547 CUBP37 71765043 IC50 = 524 nM T68547 C1UA2B 71765044 IC50 = 2700 nM T68547 C6U9VB 71769925 IC50 = 5440 nM T68547 CIRH21 71769926 IC50 = 4950 nM T68547 C26HDR 71769927 IC50 = 2370 nM T68547 C5RXY7 71769928 IC50 = 4690 nM T68547 CT1RZ2 71770054 IC50 = 20620 nM T68547 CTPJ18 71770057 IC50 = 12710 nM T68547 C1TSQ4 71770058 IC50 = 20230 nM T68547 CVU1W6 71770059 IC50 = 31380 nM T68547 CHK58Q 71770060 IC50 = 6480 nM T68547 CG3X4E 71770191 IC50 = 9660 nM T68547 CJ87KH 71770193 IC50 = 4730 nM T68547 C8J7IV 71770194 IC50 = 3420 nM T68547 CN5D6Z 71770321 IC50 = 4090 nM T68547 C13MPI 71770439 IC50 = 7880 nM T68547 C5K4ZC 71770562 IC50 = 17800 nM T68547 CTSK68 71811225 IC50 = 1880 nM T68547 C1K6OW 71811226 IC50 = 1450 nM T68547 CU3N9R 71811227 IC50 = 4890 nM T68547 CS2L4B 71811228 IC50 = 758 nM T68547 CL4DT9 71811229 IC50 = 495 nM T68547 CK6DB4 71811230 IC50 = 3200 nM T68547 CIM3G4 71811257 IC50 = 433 nM T68547 CHR8V0 71811259 IC50 = 1190 nM T68547 CVL54T 71811261 IC50 > 50000 nM T68547 CZR93K 71811262 IC50 = 2110 nM T68547 C52NYO 71811289 IC50 = 389 nM T68547 CM8BE4 71811290 IC50 = 1810 nM T68547 C0MV3O 71811291 IC50 = 18600 nM T68547 C7UYD4 71811292 IC50 = 2090 nM T68547 C7XL3N 71811293 IC50 = 48500 nM T68547 C4HBC5 71811294 IC50 = 3000 nM T68547 CTA26S 71811295 IC50 = 1940 nM T68547 CZ1P4F 71811296 IC50 = 250 nM T68547 CS0CF2 71811297 IC50 = 125 nM T68547 C6RIW8 71811298 IC50 = 114 nM T68547 C62FIE 71811300 IC50 = 182 nM T68547 C5E0DS 71811329 IC50 = 152 nM T68547 C0A3OP 71811330 IC50 = 17 nM T68547 CLTO84 71811331 IC50 = 21 nM T68547 C27AXQ 71811332 IC50 = 12 nM T68547 CBI2M7 71811333 IC50 = 80 nM T68547 CCV12Y 71811334 IC50 = 42 nM T68547 CJ23QA 71811335 IC50 = 41 nM T68547 CKC7V2 71811378 IC50 = 9.5 nM T68547 C0PRH5 71811379 IC50 = 25 nM T68547 CXVF61 71811380 IC50 = 23 nM T68547 C2WS1U 71811381 IC50 = 5.4 nM T68547 CWF49G 71811382 IC50 = 9.5 nM T68547 C6N1GC 71811383 IC50 = 5.4 nM T68547 CVS9X7 71811426 IC50 = 2.7 nM T68547 CB14VL 71811427 IC50 = 13 nM T68547 CTH41W 71811430 IC50 = 4 nM T68547 CAW2Q1 71818098 IC50 = 550 nM T68547 CT7L6G 72163687 Ki > 2500 nM T68547 CKE9D3 72163688 Ki > 2500 nM T68547 CR94ZB 72164776 Ki = 0.62 nM T68547 CI9H6L 72164895 Ki = 0.26 nM T68547 CF17AG 72164896 Ki = 0.82 nM T68547 CGPN68 72164897 Ki = 9.8 nM T68547 C6HG5M 72164898 Ki = 35 nM T68547 C7W0GL 72164899 Ki = 23 nM T68547 C64BDO 72165040 Ki = 45 nM T68547 CH68XV 72188554 IC50 = 11 nM T68547 CD17AY 72195320 IC50 = 320 nM T68547 CS5UL7 72195322 IC50 = 64 nM T68547 C6RI4C 72195326 IC50 = 2490 nM T68547 CA8D1R 72195458 IC50 = 2660 nM T68547 C0DR7G 72195459 IC50 = 233 nM T68547 CFK2Z7 72195460 IC50 = 227 nM T68547 CNJ8X0 72195461 IC50 = 376 nM T68547 CV13FT 72195463 IC50 = 539 nM T68547 CVXZ50 72195464 IC50 = 293 nM T68547 CM41HG 72195593 IC50 = 195 nM T68547 C5X2IY 72195594 IC50 = 342 nM T68547 C3N8UH 72195595 IC50 = 86 nM T68547 CIDB41 72195596 IC50 = 67 nM T68547 CQSY20 72195597 IC50 = 242 nM T68547 CO3Y1A 72195598 IC50 = 218 nM T68547 CNC56Z 72204472 IC50 = 1900 nM T68547 CR59TH 72204473 IC50 = 2750 nM T68547 CB9L8Z 72204662 IC50 = 440 nM T68547 CT7M6G 72204663 IC50 = 490 nM T68547 C1VG8U 72204664 IC50 = 250 nM T68547 CC0XI1 72204665 IC50 = 480 nM T68547 C4MW3U 72204666 IC50 = 420 nM T68547 C98VDM 72204667 IC50 = 270 nM T68547 C4FKY5 72204850 IC50 = 1090 nM T68547 CU30CD 72205221 IC50 = 700 nM T68547 C90FMR 72205411 IC50 = 550 nM T68547 CAC5Q7 72375561 IC50 = 150 nM T68547 C3WQV2 72375562 IC50 = 4.4 nM T68547 CC1W6J 72375670 IC50 = 950 nM T68547 C1A4YW 72545684 IC50 = 13 nM T68547 CY8R0O 72696205 IC50 = 14080 nM T68547 CM3KS6 72696333 IC50 = 2830 nM T68547 CI2EH8 72696334 IC50 = 590 nM T68547 C0CM8Q 72696335 IC50 = 210 nM T68547 CG31RX 72696336 IC50 = 1430 nM T68547 CJ3EH7 72696464 IC50 = 380 nM T68547 C1OA0T 72696465 IC50 = 100 nM T68547 C1I9TZ 72696466 IC50 = 243 nM T68547 CFU3V5 72696467 IC50 = 125 nM T68547 CTR52Z 72696598 IC50 = 385 nM T68547 C4O2ZT 72696599 IC50 = 93 nM T68547 C5N9BQ 72696600 IC50 = 578 nM T68547 CE87BF 72696601 IC50 = 369 nM T68547 C73XOU 72734382 IC50 = 1080 nM T68547 CJR6C9 72734542 IC50 = 370 nM T68547 CV09DJ 72734543 IC50 = 5000 nM T68547 CS6LW0 72946640 IC50 = 25 nM T68547 CXM37Z 72946641 IC50 = 43 nM T68547 CQA16N 72946833 IC50 = 34 nM T68547 CNR7Z2 72946834 IC50 = 131 nM T68547 C12JYS 72946835 IC50 = 72 nM T68547 C5Y9XH 72946836 IC50 = 33 nM T68547 CVZR94 72946837 IC50 = 1450 nM T68547 C8-AUG 72946838 IC50 = 102 nM T68547 CHQ39Y 72947043 IC50 = 59 nM T68547 CCST90 72947044 IC50 = 7 nM T68547 C7J3RH 72947045 IC50 = 32 nM T68547 CK10LZ 73292342 IC50 > 10000 nM T68547 CX3W1T 73333311 IC50 = 5800 nM T68547 C21XQI 73345596 IC50 = 40 nM T68547 C5FDJ0 73347611 IC50 > 10000 nM T68547 C68LBO 73349131 IC50 = 4 nM T68547 CN24OK 73350652 IC50 = 2180 nM T68547 CB96UM 73352206 IC50 = 67300 nM T68547 CSP58Q 73353181 IC50 = 730 nM T68547 CH6Z2L 73353182 IC50 = 850 nM T68547 C0UQO1 73353605 IC50 = 750 nM T68547 CUD02X 73355098 IC50 = 65 nM T68547 CXK86S 73355189 IC50 = 52 nM T68547 CGM2S4 73356727 IC50 > 10000 nM T68547 CVNW01 73386831 IC50 > 1000 nM T68547 C80SEC 73504974 IC50 = 2460 nM T68547 CK1BY2 73504975 IC50 = 7110 nM T68547 CE79YJ 73505176 IC50 = 5230 nM T68547 CC75WA 73505177 IC50 = 1030 nM T68547 C2LGB5 73505178 IC50 = 1950 nM T68547 CFG01S 73505179 IC50 = 2270 nM T68547 C3KVB2 73505180 IC50 = 1170 nM T68547 CNC6Q5 73505594 IC50 = 130 nM T68547 CD6L5K 73707349 IC50 = 0.7 nM T68547 C26KZD 73707535 IC50 = 2.3 nM T68547 CM1H3U 73707536 IC50 = 8 nM T68547 CH97TE 73707543 IC50 = 3.1 nM T68547 C2PWQ3 73707544 IC50 = 3.2 nM T68547 CEM5B6 73707545 IC50 = 2.1 nM T68547 CPQ43R 73707550 IC50 = 1.1 nM T68547 CJ1DA8 73774764 IC50 = 329.9 nM T68547 CQ3K6G 73776326 IC50 = 10.3 nM T68547 CC4L0G 73776327 IC50 = 13.2 nM T68547 CZB6G7 73776472 IC50 = 11.8 nM T68547 CSRE84 73776614 IC50 = 16.7 nM T68547 C01FVX 73776616 IC50 = 6 nM T68547 C3UC9H 73891099 IC50 = 8600 nM T68547 CA72JL 74221661 IC50 = 250 nM T68547 CC5GV0 74221662 IC50 = 200 nM T68547 CMU19S 74221664 IC50 = 1850 nM T68547 CT0W9Y 74221665 IC50 = 1280 nM T68547 C5F0KC 74221752 IC50 > 2500 nM T68547 C8O6HQ 74221754 IC50 = 2490 nM T68547 CS2QN0 74221755 IC50 = 2120 nM T68547 CF16BI 74221756 IC50 = 600 nM T68547 CDHA91 74221848 IC50 = 290 nM T68547 CI6YT4 74221849 IC50 = 390 nM T68547 CP16TF 74222110 IC50 = 2160 nM T68547 C9AVW2 74222111 IC50 = 340 nM T68547 C7X6GT 76311016 IC50 = 336.6 nM T68547 CM6H9C 76324878 IC50 = 22000 nM T68547 CL4JQ3 76331862 IC50 = 1790 nM T68547 CTZ53J 76332759 IC50 = 0.2 nM T68547 C08CPW 76335428 IC50 = 77 nM T68547 CKI74A 76853213 IC50 = 4300 nM T68547 C0ZKI5 76853285 IC50 = 15 nM T68547 CCR7L2 76853289 IC50 > 100000 nM T68547 C96LMJ 78323868 IC50 = 35 nM T68547 C5IAU4 78323870 IC50 = 28 nM T68547 CJ6Z0X 78324068 IC50 > 20000 nM T68547 C25ETN 78324161 IC50 = 63 nM T68547 C3U0KE 81689842 IC50 = 39700 nM T68547 CG5ZD9 86291495 IC50 = 3.8 nM T68547 C61VCD 86294741 IC50 = 270000 nM T68547 CBWV30 86294747 IC50 = 93000 nM T68547 CGF12C 86302517 IC50 = 49 nM T68547 C8O5PZ 86302518 IC50 = 36 nM T68547 CL78UP 86302519 IC50 = 57 nM T68547 CY5Q0E 86302520 IC50 = 50 nM T68547 C06YBD 86302594 IC50 = 2030 nM T68547 CQ1OA0 86342535 IC50 = 48 nM T68547 C3EM7H 86581004 IC50 = 24 nM T68547 C7UK3Y 86581005 IC50 = 30 nM T68547 CY64UM 86581152 IC50 = 14 nM T68547 CY5V7C 86581153 IC50 = 9.1 nM T68547 C1HE8I 86581432 IC50 = 670 nM T68547 CZM07I 86581434 IC50 = 66 nM T68547 C8ZQG9 86581435 IC50 = 35 nM T68547 C6M9PL 86765212 IC50 = 310 nM T68547 CS5I4Y 87261507 IC50 = 70 nM T68547 CK5B2E 87290521 IC50 = 0.6 nM T68547 C4BGX3 87290562 IC50 = 0.8 nM T68547 CXD9F5 87290634 IC50 = 0.9 nM T68547 CP1CQ9 87331876 IC50 = 1.4 nM T68547 C5JIT0 87618609 IC50 = 5600 nM T68547 CRQO37 88005144 IC50 = 800 nM T68547 CRAX13 88849486 IC50 = 11700 nM T68547 CD3X6M 88849490 IC50 = 19500 nM T68547 CQ2LF5 88920533 IC50 = 9730 nM T68547 CP1NA9 89183138 IC50 = 72 nM T68547 CQS6C0 89183185 IC50 = 123 nM T68547 CB47VC 89464167 IC50 = 1750 nM T68547 CR27YF 89827822 IC50 = 5740 nM T68547 C82QNF 90149109 IC50 > 5000 nM T68547 CUBX58 90149126 IC50 > 5000 nM T68547 C86IMD 90149143 IC50 = 2620 nM T68547 CGBD45 90149248 IC50 > 5000 nM T68547 CVOM90 90149517 IC50 > 2500 nM T68547 C2CE9A 90643781 IC50 = 14 nM T68547 C05MTO 90643782 IC50 = 20 nM T68547 C6RM2B 90643783 IC50 = 18 nM T68547 CPD10X 90643784 IC50 = 51 nM T68547 CUB0Q1 90643785 IC50 = 580 nM T68547 C43MQN 90644925 IC50 = 16820 nM T68547 CDM3H5 90644926 IC50 = 13860 nM T68547 CD7J6C 90644927 IC50 = 170 nM T68547 C62GSL 90654859 IC50 = 355.4 nM T68547 CYW51P 90654946 IC50 = 48500 nM T68547 CJH1S6 90654947 IC50 = 60100 nM T68547 CSR56C 90655296 IC50 = 3100 nM T68547 C15WHB 90656724 IC50 = 4850 nM T68547 CSDO81 90664458 Ki = 28 nM T68547 CI9M0E 90665809 IC50 = 0.48 nM T68547 C23GNF 90665810 IC50 = 0.94 nM T68547 CY0P7X 90665811 IC50 = 2.6 nM T68547 C0RX4B 90667452 IC50 = 250 nM T68547 C8HL5V 90667453 IC50 = 250 nM T68547 C3IE7F 90667454 IC50 = 50 nM T68547 C37GOB 90667455 IC50 = 900 nM T68547 C67UHD 91619090 IC50 = 25000 nM T68547 C6JZT7 91619093 IC50 = 29870 nM T68547 CAQL21 91667420 IC50 = 42 nM T68547 C5M9AK 91667421 IC50 = 13.2 nM T68547 CJO6T1 91810840 IC50 = 800 nM T68547 CYJ12Q 91884636 IC50 = 13 nM T68547 CTUB92 91900719 IC50 = 260 nM T68547 C0FCU9 91938063 IC50 = 26.28 nM T68547 C34WIG 92045024 IC50 = 6310 nM T68547 CN5KS8 92135978 IC50 = 4600 nM T68547 CJQK17 101068910 IC50 = 3 nM T68547 CYO9J5 101879983 IC50 = 1.14 nM T68547 C9OC0F 101882265 IC50 = 21300 nM T68547 C2I8XR 101882814 Ki = 2400 nM T68547 CVE07R 101882857 IC50 = 373 nM T68547 C63EWT 101882858 IC50 = 1260 nM T68547 C8KZB4 101883993 Ki = 600 nM T68547 C7Q6ID 101884982 IC50 = 24 nM T68547 CR46PQ 101884983 IC50 = 10 nM T68547 CRZ83C 101884989 IC50 = 101 nM T68547 C7PS2E 102140473 IC50 = 13.9 nM T68547 C3PFY8 102140474 IC50 = 27 nM T68547 C12GJX 102366363 IC50 = 200 nM T68547 CO25LD 102366364 IC50 = 200 nM T68547 C8CER4 102366365 IC50 = 200 nM T68547 CT7Z8F 102514716 IC50 > 10000 nM T68547 CS2UL0 117829456 IC50 = 52 nM T68547 C7L4OT 117829461 IC50 = 43 nM T68547 C50VUN 117829462 IC50 = 89 nM T68547 CPW71E 117855070 IC50 = 604 nM T68547 CB68IV 117855071 IC50 = 721 nM T68547 CW61HU 118453221 IC50 = 1760 nM T68547 CH27PR 118613747 IC50 = 5.5 nM T68547 C0OX4M 118613748 IC50 = 0.62 nM T68547 CNF09H 118613750 IC50 = 39 nM T68547 C3ETI2 118613751 IC50 = 2.3 nM T68547 C9KZQ0 118613755 IC50 = 0.2 nM T68547 C30OPU 118613756 IC50 = 3.3 nM T68547 C46TFD 118613757 IC50 = 0.96 nM T68547 C1J5AG 118613783 IC50 = 0.29 nM T68547 C9T0ML 118613821 IC50 = 0.21 nM T68547 CSU52M 118656852 IC50 = 9400 nM T68547 CB6AJ9 118656853 IC50 = 12000 nM T68547 CK6YX4 118706143 IC50 = 31 nM T68547 C8JMF2 118706144 IC50 = 25 nM T68547 CZY1Q2 118706145 IC50 = 25 nM T68547 CC3LG6 118706146 IC50 = 37 nM T68547 CVCM47 118706554 IC50 = 12.7 nM T68547 C98SPM 118706555 IC50 = 8.1 nM T68547 CB8Q2L 118706556 IC50 = 4.9 nM T68547 CV3ST1 118706557 IC50 = 16 nM T68547 CAF41G 118707835 IC50 = 800 nM T68547 C0P4EV 118707836 IC50 = 600 nM T68547 CC8KL3 118707837 IC50 = 9900 nM T68547 C9VI8U 118707838 IC50 = 1000 nM T68547 CRU9G3 118707839 IC50 = 2400 nM T68547 C9SWI4 118707840 IC50 = 1500 nM T68547 CW9UJ1 118707841 IC50 = 4100 nM T68547 CBYI69 118707842 IC50 = 300 nM T68547 C45UYG 118709095 IC50 = 59000 nM T68547 C7QHE4 118712502 IC50 = 0.3 nM T68547 C8KSD6 118712503 IC50 = 0.4 nM T68547 C5SP1G 118714365 IC50 = 191 nM T68547 CA09PT 118714366 IC50 = 367 nM T68547 CTZ2Q1 118714367 IC50 = 266 nM T68547 CW3Y7E 118714368 IC50 = 35 nM T68547 C1GC6I 118714369 IC50 = 1160 nM T68547 C2NR1W 118714370 IC50 = 1760 nM T68547 C1JFZ7 118714371 IC50 = 313 nM T68547 CIC8A7 118714372 IC50 = 1310 nM T68547 C5QD4H 118714373 IC50 = 323 nM T68547 CM27KC 118714374 IC50 = 197 nM T68547 CXF0U3 118714375 IC50 = 75 nM T68547 C2M5OR 118714376 IC50 = 35 nM T68547 CY4GN9 118714377 IC50 = 33 nM T68547 C86WSR 118714378 IC50 = 145 nM T68547 CKWQ53 118714379 IC50 = 719 nM T68547 C2W0KJ 118714380 IC50 = 68 nM T68547 CL3ZF9 118714381 IC50 = 116 nM T68547 CMJF26 118714382 IC50 = 43 nM T68547 CV04TX 118714383 IC50 = 646 nM T68547 C8LVO5 118714384 IC50 = 202 nM T68547 CER3U4 118714385 IC50 = 9580 nM T68547 CDL25Z 118714411 IC50 = 15700 nM T68547 CVZ78U 118714412 IC50 = 900 nM T68547 COR95F 118714413 IC50 = 8900 nM T68547 CRL92Y 118714414 IC50 = 800 nM T68547 CR37MV 118714415 IC50 = 2100 nM T68547 C96XGO 118715268 IC50 = 11200 nM T68547 C7P3KH 118715726 IC50 = 131.3 nM T68547 CK6UM0 118715727 IC50 = 35.89 nM T68547 CW85VZ 118715728 IC50 = 13.36 nM T68547 C39EXL 118715729 IC50 = 218.1 nM T68547 CYGT73 118715730 IC50 = 40.84 nM T68547 CCAM49 118715731 IC50 = 21.67 nM T68547 C37NXA 118715732 IC50 = 10.07 nM T68547 CEN1J3 118715733 IC50 = 12.5 nM T68547 CFD2B8 118715734 IC50 = 13.54 nM T68547 CO8TJ6 118715735 IC50 = 6.24 nM T68547 C90TIX 118715736 IC50 = 7.78 nM T68547 C14KQU 118715737 IC50 = 3.24 nM T68547 CMK8B7 118715738 IC50 = 11.77 nM T68547 CQ6V9M 118715739 IC50 = 1.9 nM T68547 CWM04T 118715740 IC50 = 14.01 nM T68547 CLYS39 118715741 IC50 = 2.01 nM T68547 C04XZU 118715742 IC50 = 29.82 nM T68547 CJ4FS3 118715743 IC50 = 32.87 nM T68547 C3BH1K 118715744 IC50 = 4.57 nM T68547 CA12OP 118715745 IC50 = 4.51 nM T68547 C51RTI 118715746 IC50 = 2.97 nM T68547 CFX16A 118715747 IC50 = 5.39 nM T68547 C5OWL1 118715748 IC50 = 14.49 nM T68547 C8AW9X 118715749 IC50 = 13.85 nM T68547 C2Y7ZC 118715750 IC50 = 25.53 nM T68547 CM5QT7 118719376 Ki = 1200 nM T68547 CPB7C3 118719377 Ki = 700 nM T68547 C09OGH 118719378 Ki = 500 nM T68547 CR5VC1 118719379 Ki = 900 nM T68547 C32LCM 118719380 Ki = 1000 nM T68547 C8U6YR 118719381 Ki = 900 nM T68547 C9Y0HV 118719382 Ki = 300 nM T68547 CY0J4D 118719383 Ki = 200 nM T68547 CCYU59 118719817 IC50 = 5 nM T68547 CSC47W 118720522 IC50 = 219.1 nM T68547 CUI51W 118720529 IC50 = 33.2 nM T68547 CCGH73 118720703 IC50 = 21000 nM T68547 C1EC5S 118721286 IC50 = 43 nM T68547 CMV2W9 118721625 IC50 = 7 nM T68547 CF5TO3 118721859 IC50 = 58 nM T68547 CK97TZ 118721860 IC50 = 5 nM T68547 CYV30O 118721861 IC50 = 4 nM T68547 C5WYI1 118721862 IC50 = 3 nM T68547 CSMW25 118721863 IC50 = 865 nM T68547 C5B1KM 118721864 IC50 = 160 nM T68547 CG8LZ0 118721865 IC50 = 5960 nM T68547 CPCN23 118721866 IC50 = 3160 nM T68547 CM0A9U 118721867 IC50 = 3210 nM T68547 CN47HE 118733259 IC50 > 100000 nM T68547 CJLN15 118733260 IC50 > 100000 nM T68547 CU8T7G 118733373 IC50 = 29400 nM T68547 C6OEU2 118733374 IC50 = 74100 nM T68547 CW5JY8 118733375 IC50 = 24500 nM T68547 C8IAG9 118734664 IC50 = 15920 nM T68547 CJ6KL7 118734665 IC50 = 2240 nM T68547 C2VQ5P 118734666 IC50 = 9620 nM T68547 CYF71E 118734667 IC50 = 1500 nM T68547 CQC7H0 118734668 IC50 = 12500 nM T68547 CP27CN 118734669 IC50 = 3320 nM T68547 CBIY72 118734670 IC50 > 20 ug.mL-1 T68547 C9C7UX 118734705 IC50 = 25500 nM T68547 C16OUT 118735146 IC50 = 280 nM T68547 CZRV81 118735147 IC50 = 210 nM T68547 CFE4D0 118735148 IC50 = 180 nM T68547 C97NHV 118735149 IC50 = 2750 nM T68547 CQ0FJ3 118735150 IC50 = 90 nM T68547 CD4J8E 118735151 IC50 = 60 nM T68547 C7UE8T 118735152 IC50 = 110 nM T68547 CS6WO5 118735153 IC50 = 3850 nM T68547 C4XZ3C 118735154 IC50 = 5260 nM T68547 CRL6V4 118735155 IC50 = 70 nM T68547 CI8G4X 118737400 IC50 = 1420 nM T68547 C2F8TQ 118737455 IC50 = 241 nM T68547 C1T6WZ 118738004 IC50 > 10000 nM T68547 CZ61KV 118753026 IC50 = 140 nM T68547 CFI23Y 118753027 IC50 = 970 nM T68547 C75LTK 118753189 IC50 = 4600 nM T68547 CM3FB8 118796366 IC50 = 33600 nM T68547 C5L8QM 118884518 IC50 = 8450 nM T68547 CB84TO 121278998 IC50 > 50000 nM T68547 C9S5OK 121279020 IC50 > 50000 nM T68547 CVXA98 121304930 IC50 >= 10000 nM T68547 CIA40K 121472983 IC50 > 10000 nM T68547 CL3M2F 121499152 Ki = 176 nM T68547 C93JAV 122177622 IC50 = 371 nM T68547 C5HJ0C 122177623 IC50 > 10000 nM T68547 CT9M7U 122177954 IC50 = 30 nM T68547 COJ4I8 122177955 IC50 = 321 nM T68547 C5R2AU 122177956 IC50 = 190 nM T68547 CSU97K 122177957 IC50 = 24 nM T68547 C0OGM1 122177958 IC50 > 10000 nM T68547 CP5F3X 122177959 IC50 = 93 nM T68547 CO9QK7 122177960 IC50 = 89 nM T68547 CL1X2G 122177961 IC50 = 527 nM T68547 C4DR1I 122177962 IC50 = 275 nM T68547 CUY18X 122177966 IC50 > 10000 nM T68547 CNY91L 122177967 IC50 = 64 nM T68547 CR8WL1 122180003 IC50 > 10000 nM T68547 CRW9F3 122180812 IC50 = 534 nM T68547 CJ42OQ 122180814 IC50 = 107 nM T68547 CEW23B 122180816 IC50 = 583 nM T68547 CBO5T8 122180819 IC50 = 2980 nM T68547 CC80JD 122180822 IC50 = 22 nM T68547 CYCT17 122180828 IC50 = 241 nM T68547 CL16JS 122180834 IC50 = 282 nM T68547 CYD03G 122181048 IC50 = 349 nM T68547 CIZX38 122181808 IC50 = 118 nM T68547 CE8OF0 122181809 IC50 = 154 nM T68547 COPU35 122181810 IC50 = 129 nM T68547 CX21ZC 122181811 IC50 = 217 nM T68547 CB2T9X 122181812 IC50 = 173 nM T68547 CW92GL 122181813 IC50 = 178 nM T68547 C1QKZ4 122181814 IC50 = 120 nM T68547 CX8M2E 122181815 IC50 = 169 nM T68547 CCK65N 122181816 IC50 = 131 nM T68547 CMBI41 122181817 IC50 = 137 nM T68547 CW4K2U 122181880 IC50 = 203.6 nM T68547 CK63UH 122181881 IC50 = 340 nM T68547 C0H9WU 122181882 IC50 = 2.2 nM T68547 CR3TU6 122181883 IC50 = 340.3 nM T68547 C57VRL 122181884 IC50 = 816.9 nM T68547 C81QDF 122182040 IC50 = 201.16 nM T68547 C2VO8E 122184845 IC50 = 15.46 nM T68547 CGSF80 122184846 IC50 = 17.47 nM T68547 CN4H8Q 122184847 IC50 = 4.17 nM T68547 CT94PN 122184848 IC50 = 5.75 nM T68547 CI2X8M 122184849 IC50 = 35.41 nM T68547 C5HOK3 122184850 IC50 = 19.49 nM T68547 CZC3Q4 122184851 IC50 = 15.43 nM T68547 CQW6T3 122184852 IC50 = 17.98 nM T68547 CE4M7C 122184853 IC50 = 263 nM T68547 C7MT9U 122184854 IC50 = 45.85 nM T68547 C4AQ5H 122184855 IC50 = 41.63 nM T68547 C07UQJ 122184856 IC50 = 27.91 nM T68547 CST56N 122184857 IC50 = 65.77 nM T68547 C6K1HJ 122184858 IC50 = 68.98 nM T68547 CG19IO 122185146 IC50 = 66.02 nM T68547 CI4U2H 122185147 IC50 = 98.08 nM T68547 CU47DI 122185148 IC50 = 272.08 nM T68547 C9XMU5 122185149 IC50 = 323.23 nM T68547 C5QCF0 122185150 IC50 = 205.34 nM T68547 CSA1H8 122185151 IC50 = 570.99 nM T68547 CZG70W 122185152 IC50 = 439.06 nM T68547 C9V6XI 122186483 IC50 = 240 nM T68547 CU74JP 122186484 IC50 = 380 nM T68547 C7M2EU 122186485 IC50 = 1200 nM T68547 CI32QY 122186544 IC50 = 700 nM T68547 CBN3P1 122186553 IC50 = 76 nM T68547 CP83NA 122186554 IC50 = 390 nM T68547 CRTN32 122191260 IC50 = 1310 nM T68547 C28JVO 122192004 IC50 = 2.18 nM T68547 CF2D8U 122192005 IC50 = 165 nM T68547 CV8YH0 122193364 IC50 = 1270 nM T68547 C1CI0Z 122193365 IC50 = 820 nM T68547 C32LTK 122193367 IC50 = 1050 nM T68547 CE04LR 122193368 IC50 = 1040 nM T68547 CW1HK5 122195536 IC50 = 3.5 nM T68547 C5W8OZ 122376192 IC50 = 5.25 nM T68547 C2YLS8 122379529 IC50 = 83.22 nM T68547 CCI4M6 122379531 IC50 = 66.83 nM T68547 CZ74QC 122379532 IC50 = 64.7 nM T68547 CLZ19M 122379533 IC50 = 203.71 nM T68547 CL0X8K 122550124 IC50 > 1000 nM T68547 C24QLO 122550126 IC50 = 272 nM T68547 CNKM78 122550129 IC50 = 76 nM T68547 CL31AN 122550132 IC50 = 242 nM T68547 CJM9X5 122550134 IC50 = 203 nM T68547 CHS4F7 122550135 IC50 = 176 nM T68547 CB8J6A 122550165 IC50 > 1000 nM T68547 CZ6TC9 122550171 IC50 > 1000 nM T68547 CX87LD 122550174 IC50 = 253 nM T68547 C3V5ND 122550211 IC50 = 422 nM T68547 C64OME 122550212 IC50 = 84 nM T68547 C8PM6C 122550213 IC50 = 160 nM T68547 CAXY60 122550234 IC50 = 172 nM T68547 CAOH68 122550235 IC50 = 204 nM T68547 CR38WT 122550251 IC50 = 73 nM T68547 CX61TL 122550293 IC50 = 306 nM T68547 C63EYP 122601008 IC50 > 3000 nM T68547 CCN03D 122601010 IC50 > 10000 nM T68547 CZC01M 122601076 IC50 > 3000 nM T68547 C6Z5WJ 122648316 IC50 = 62 nM T68547 CX46DA 122648323 IC50 = 1.6 nM T68547 CI1AJ9 122648339 IC50 = 1.02 nM T68547 CZE35C 122648343 IC50 = 0.45 nM T68547 C7UYV1 122648344 IC50 = 1 nM T68547 C71PAY 122648346 IC50 = 0.55 nM T68547 C8J4FT 122648347 IC50 = 1.59 nM T68547 CE5Z0G 122648364 IC50 = 110 nM T68547 CMPQ34 122648365 IC50 = 125 nM T68547 C58IPE 122648366 IC50 = 0.97 nM T68547 C54RNT 122648367 IC50 = 0.65 nM T68547 C0IBF7 122648403 IC50 = 0.49 nM T68547 C8MO7V 122648552 IC50 = 1.1 nM T68547 C3AKB1 122648553 IC50 = 5.1 nM T68547 C9WQ1N 122648555 IC50 = 0.81 nM T68547 CF0RM9 122648559 IC50 = 0.85 nM T68547 CI61WJ 122648563 IC50 = 10.01 nM T68547 C4PZ1A 122648565 IC50 = 1 nM T68547 CE19SM 122648568 IC50 = 30.1 nM T68547 CBTO34 122648569 IC50 = 6.15 nM T68547 CA7L8O 122648570 IC50 = 1.01 nM T68547 CM3O4F 122648571 IC50 = 1.98 nM T68547 CY6BO5 122648574 IC50 = 1.1 nM T68547 CPDN98 122648575 IC50 = 1.11 nM T68547 CX7ZC1 122648576 IC50 = 1.14 nM T68547 C1UVI7 122648600 IC50 = 1 nM T68547 C69KVZ 122648605 IC50 = 10 nM T68547 CI4EB6 122648645 IC50 = 1.6 nM T68547 C8HG7U 122648646 IC50 = 67 nM T68547 CMX59K 122648648 IC50 = 1.04 nM T68547 CVZ64I 122648649 IC50 = 0.55 nM T68547 CW03VD 126582837 IC50 = 66.09 nM T68547 C5UV6J 126582839 IC50 = 33.6 nM T68547 CR9AC4 126582841 IC50 = 97.28 nM T68547 C1HS3A 126582843 IC50 = 19.38 nM T68547 CFI58L 126582907 IC50 = 159.55 nM T68547 CMT02Y 126582908 IC50 = 9750.65 nM T68547 C6W3RK 126648983 IC50 = 436 nM T68547 CTP62U 126649182 IC50 = 16900 nM T68547 CM6YJ3 126649211 IC50 = 307 nM T68547 CZ67DK 126738293 IC50 = 7490 nM T68547 CEC14P 126738294 IC50 = 6880 nM T68547 C59SEH 126738297 IC50 > 30000 nM T68547 CLO14J 126738589 IC50 = 6570 nM T68547 C3Q6FV 127024856 IC50 = 2200 nM T68547 CVFI87 127025051 IC50 > 10000 nM T68547 CQ39UE 127025078 IC50 = 40070 nM T68547 C8FOZ4 127025172 IC50 > 10000 nM T68547 CE4CI8 127025178 IC50 = 52 nM T68547 CL8TF5 127025475 IC50 > 10000 nM T68547 C8VEY9 127025539 IC50 > 10000 nM T68547 CNSO40 127025540 IC50 = 850 nM T68547 CM38EU 127025541 IC50 = 21 nM T68547 CY5T9P 127025646 IC50 > 3000 nM T68547 CKJ6L8 127025647 IC50 > 3000 nM T68547 CXVC21 127025656 IC50 = 19560 nM T68547 CF4G7Q 127025769 IC50 > 10000 nM T68547 CIF74W 127025777 IC50 > 10000 nM T68547 CT2EK9 127025778 IC50 > 10000 nM T68547 CMWO84 127025780 IC50 > 10000 nM T68547 CWB73C 127025940 IC50 = 33450 nM T68547 C58JDE 127025947 IC50 = 14870 nM T68547 CQ32BA 127026381 IC50 > 10000 nM T68547 CQTF36 127026436 IC50 > 10000 nM T68547 C3Q8FL 127026437 IC50 > 10000 nM T68547 C2N1UD 127026438 IC50 > 10000 nM T68547 CWY63G 127026695 IC50 = 526 nM T68547 CO4JI5 127026735 IC50 = 220 nM T68547 CME4B7 127026736 IC50 = 650 nM T68547 CG34KC 127026737 IC50 = 130 nM T68547 CNX10Q 127026738 IC50 = 1300 nM T68547 CJ0AI5 127026739 IC50 = 250 nM T68547 C60DIS 127026740 IC50 > 10000 nM T68547 C31UJC 127026741 IC50 > 10000 nM T68547 COI3S8 127026742 IC50 = 1900 nM T68547 CCR4M7 127026743 IC50 = 2700 nM T68547 CNH5P8 127026863 IC50 = 83580 nM T68547 C0BG8P 127027017 IC50 = 225 nM T68547 C1R4SF 127027021 IC50 = 331 nM T68547 CZR43H 127027067 IC50 = 1800 nM T68547 CA1N7Y 127027068 IC50 = 3300 nM T68547 CE8CN3 127027069 IC50 = 3600 nM T68547 CCG30L 127027070 IC50 = 440 nM T68547 CU84JL 127027071 IC50 > 10000 nM T68547 CSJ18X 127027150 IC50 = 22470 nM T68547 CA58GI 127027171 IC50 = 14470 nM T68547 CBT4S5 127027172 IC50 = 22630 nM T68547 C3UED2 127027173 IC50 = 23750 nM T68547 CUSY71 127027174 IC50 = 32890 nM T68547 C2OIE1 127027175 IC50 = 12210 nM T68547 CT5VX3 127027322 IC50 > 10000 nM T68547 CJAE38 127027376 IC50 > 10000 nM T68547 C86OFN 127027393 IC50 > 10000 nM T68547 C8X6FT 127027394 IC50 > 10000 nM T68547 CK0J7H 127027395 IC50 > 10000 nM T68547 CTP3J4 127027396 IC50 > 10000 nM T68547 COU4I9 127027458 IC50 = 93890 nM T68547 CC0WJ2 127027462 IC50 = 36510 nM T68547 CSZL73 127027477 IC50 = 17460 nM T68547 CY3P7V 127027483 IC50 = 19080 nM T68547 C68TYH 127027490 IC50 = 3480 nM T68547 CA14VM 127027506 IC50 = 1843.92 nM T68547 CB9PL5 127027507 IC50 > 10000 nM T68547 CBOJ07 127027508 IC50 > 10000 nM T68547 CT18SH 127027509 IC50 > 10000 nM T68547 CJ8MQ3 127027677 IC50 = 98 nM T68547 C3EWH4 127027679 IC50 = 310 nM T68547 C1KWD3 127027680 IC50 = 422 nM T68547 CM3SZ5 127027716 IC50 = 2300 nM T68547 CM42UC 127027717 IC50 = 1400 nM T68547 CBMZ67 127027718 IC50 > 10000 nM T68547 C1KVR2 127027719 IC50 > 10000 nM T68547 CD4T1B 127027794 IC50 = 47660 nM T68547 CG7Q3V 127027808 IC50 = 25100 nM T68547 C6JUF9 127027813 IC50 > 30000 nM T68547 CW8F7D 127027975 IC50 = 2100 nM T68547 C2QYV5 127027979 IC50 = 330 nM T68547 CX80AH 127027993 IC50 = 429 nM T68547 CO5E1V 127027994 IC50 = 133 nM T68547 CG8NU7 127027995 IC50 = 12 nM T68547 CZ7C3D 127028030 IC50 = 1.8 nM T68547 CLN54U 127028295 IC50 = 578 nM T68547 CL7EN6 127028391 IC50 = 29480 nM T68547 CG91JU 127028631 IC50 > 10000 nM T68547 CW04XE 127028723 IC50 = 10270 nM T68547 CV07OM 127028943 IC50 = 15 nM T68547 C08RCM 127028973 IC50 = 124 nM T68547 C8FNI2 127029515 IC50 > 10000 nM T68547 CV9I8D 127030313 IC50 = 5400 nM T68547 CN6K5P 127030500 IC50 = 212 nM T68547 CCNK89 127030846 IC50 > 1000 nM T68547 CI8WG4 127031734 IC50 = 195 nM T68547 C40HQA 127031756 IC50 = 264 nM T68547 C9Q1WD 127031757 IC50 = 120 nM T68547 CD1TP7 127034929 IC50 > 10000 nM T68547 CU1M3B 127034930 IC50 > 10000 nM T68547 C4SI0Q 127034947 IC50 > 10000 nM T68547 CMS1F6 127034948 IC50 = 269 nM T68547 C3VB0I 127034949 IC50 = 73.1 nM T68547 CQC2F9 127035098 IC50 = 109 nM T68547 CBP64A 127035107 IC50 = 54.5 nM T68547 CAXL98 127035256 IC50 > 10000 nM T68547 CBJG94 127035257 IC50 > 10000 nM T68547 C29AJN 127035766 IC50 = 20.8 nM T68547 C4GI0F 127037614 IC50 = 82 nM T68547 C18FSM 127039340 IC50 = 26 nM T68547 CIO0G3 127039341 IC50 = 79 nM T68547 C12NJF 127039347 IC50 = 240 nM T68547 CZ8A1F 127041696 IC50 = 30560 nM T68547 C69IXG 127041845 IC50 = 110 nM T68547 C5D2OJ 127044292 IC50 = 1430 nM T68547 C58KRZ 127044343 IC50 = 1220 nM T68547 C1TYS6 127044344 IC50 = 45 nM T68547 CJZ5M6 127044418 IC50 = 23940 nM T68547 CI65UA 127044427 IC50 > 2500 nM T68547 C3G0SM 127044498 IC50 = 467 nM T68547 CVHA97 127044853 IC50 = 240 nM T68547 C3O4VS 127044854 IC50 = 300 nM T68547 CBM5H4 127045160 IC50 = 1.37 nM T68547 C6O8FN 127045161 IC50 = 165 nM T68547 C49IGC 127045162 IC50 = 190 nM T68547 CM5B0U 127045163 IC50 = 2.62 nM T68547 C5CP9M 127045259 IC50 = 5590 nM T68547 CO72YC 127045674 IC50 = 2700 nM T68547 CTG0U3 127045675 IC50 = 6300 nM T68547 CD42EQ 127045676 IC50 = 2600 nM T68547 C9K0TN 127045677 IC50 = 2900 nM T68547 CK51QO 127045678 IC50 = 13000 nM T68547 C0HQZ3 127046055 IC50 = 129900 nM T68547 CG13WB 127046056 IC50 = 42300 nM T68547 CIQA39 127046057 IC50 = 8400 nM T68547 CC89WM 127046659 IC50 = 2400 nM T68547 CR61BE 127046852 IC50 = 31600 nM T68547 CXJM94 127046853 IC50 = 2080 nM T68547 C42VYT 127046854 IC50 = 12100 nM T68547 CR6AH4 127046855 IC50 = 20000 nM T68547 CM76WI 127046917 IC50 = 7400 nM T68547 CQ8LT6 127047324 IC50 = 3800 nM T68547 CJ7YR6 127047335 IC50 = 4100 nM T68547 CB0O4H 127047412 IC50 = 4400 nM T68547 C5OH2V 127047413 IC50 = 28900 nM T68547 CEUB27 127047550 IC50 = 9400 nM T68547 CU1M3Q 127047551 IC50 = 6400 nM T68547 CKH4S0 127047552 IC50 = 8500 nM T68547 C7TV8A 127047636 IC50 = 9600 nM T68547 C4N2BY 127047651 IC50 = 2300 nM T68547 C5SW8E 127047652 IC50 = 22300 nM T68547 CE1K8N 127047653 IC50 = 11600 nM T68547 C2KB3W 127048062 IC50 = 3600 nM T68547 CD2T1E 127051228 IC50 = 760 nM T68547 CPS8R6 127051229 IC50 = 270 nM T68547 CRZ3A6 127051526 IC50 = 150 nM T68547 CR0P6Q 127051527 IC50 = 360 nM T68547 C9V3AX 127052165 IC50 = 5450 nM T68547 C2OHP4 127052166 IC50 = 1490 nM T68547 CS60GZ 127052167 IC50 = 1430 nM T68547 C2RB3T 127052469 IC50 = 1740 nM T68547 CHA05V 127052470 IC50 = 970 nM T68547 CB8HR2 129104138 IC50 > 50000 nM T68547 CCH65A 129104183 IC50 > 50000 nM T68547 CFH8Q4 129104227 IC50 > 50000 nM T68547 C6HM5P 129104349 IC50 > 50000 nM T68547 CZTF90 129104374 IC50 > 50000 nM T68547 CUJ2P5 129104402 IC50 > 50000 nM T68547 CY3I6X 129104426 IC50 > 50000 nM T68547 C8IEV4 130258911 IC50 = 1055 nM T68547 CUYQ28 130345472 IC50 = 5230 nM T68547 CHVF85 132022730 IC50 = 33000 nM T68547 C6OXE3 132134663 IC50 = 222 nM T68547 CP8L7V 132137973 IC50 = 1436 nM T68547 C6X3HG 132145728 IC50 = 7050 nM T68547 C8O9DP 132157820 IC50 = 9550 nM T68547 C2N5JD 132279660 IC50 = 260 nM T68547 C0G9TV 132495274 IC50 = 0.72 nM T68547 COVK82 132515050 IC50 = 270 nM T68547 CJ25PE 132515051 IC50 = 80 nM T68547 C4L6UZ 132547258 IC50 = 261 nM T68547 CGBR54 132547259 IC50 = 1030 nM T68547 CW4MP2 132547260 IC50 = 980 nM T68547 C1YO2Z 132547261 IC50 = 89 nM T68547 CXT18G 132559046 IC50 = 37 nM T68547 C7C8AK 132559047 IC50 = 17 nM T68547 CAE84Z 132559048 IC50 = 530 nM T68547 CNM7O5 132559049 IC50 = 29 nM T68547 CU63DV 132569672 IC50 = 32 nM T68547 C1OJM4 132576507 IC50 = 38.25 nM T68547 CRQ0L4 132576509 IC50 = 502.8 nM T68547 CIUZ08 132576538 IC50 = 232 nM T68547 CTE3A6 132576539 IC50 = 128 nM T68547 C87DPY 132576540 IC50 = 179 nM T68547 CG91UP 132576541 IC50 = 366 nM T68547 CL2R5W 132576542 IC50 = 288 nM T68547 C5C2EQ 132576544 IC50 = 448 nM T68547 CA5V0R 132576546 IC50 = 742 nM T68547 CEH95L 132576588 IC50 > 10000 nM T68547 C0Y2TP 132585192 IC50 = 25 nM T68547 C0Z2PH 132850192 IC50 = 3700 nM T68547 C4KE3N 132938351 IC50 = 415 nM T68547 C4UAN3 134129876 IC50 = 208 nM T68547 C25EVA 134129883 IC50 = 111 nM T68547 CWRH43 134129994 IC50 = 400 nM T68547 CK2TM6 134130010 IC50 = 1870 nM T68547 CYW6H1 134130165 IC50 = 60 nM T68547 C8CY7S 134131006 IC50 = 1760 nM T68547 CQ7SN8 134131102 IC50 = 968 nM T68547 CYCS54 134131113 IC50 = 1810 nM T68547 CQO23I 134131456 IC50 = 251 nM T68547 CHZ8A3 134131564 IC50 = 778 nM T68547 CN9DL4 134132030 IC50 > 10000 nM T68547 CA7J2D 134132574 IC50 = 8.3 nM T68547 CDMJ75 134135414 IC50 = 5.6 nM T68547 CX93QK 134135812 IC50 > 100000 nM T68547 CN8L9J 134136160 IC50 = 330000 nM T68547 CA5P7T 134136358 IC50 = 973.1 nM T68547 C53UTO 134137062 IC50 = 3150 nM T68547 CYGZ85 134137500 IC50 = 5.2 nM T68547 CJC1E8 134137789 IC50 = 6.9 nM T68547 C3RA6C 134138227 IC50 = 1.4 nM T68547 CSX58U 134139437 IC50 > 10000 nM T68547 CK7EZ2 134139706 IC50 = 26.6 nM T68547 CCF0X1 134140501 IC50 = 7 nM T68547 C08YTI 134140697 IC50 = 5.74 nM T68547 C75NRQ 134141877 IC50 > 100000 nM T68547 C62SVR 134142119 IC50 > 100000 nM T68547 CLI48U 134143743 IC50 = 6190 nM T68547 CUA26W 134143927 IC50 = 48000 nM T68547 CEDU72 134145690 IC50 = 2340 nM T68547 C1E2ZW 134145921 IC50 = 2400 nM T68547 CWRJ15 134147087 IC50 > 100000 nM T68547 C8K0XJ 134147090 IC50 > 10000 nM T68547 C8O9SN 134147898 IC50 = 4070 nM T68547 CP14DK 134149339 IC50 = 7.2 nM T68547 CQ61SB 134150479 IC50 = 58100 nM T68547 CM7H0R 134150543 IC50 = 38.6 nM T68547 CJX12K 134151832 IC50 = 3090 nM T68547 CDX75O 134152551 IC50 = 20600 nM T68547 C2JV5X 134153768 IC50 > 100000 nM T68547 C2E8MV 134154228 IC50 = 14 nM T68547 CBY2R8 134156011 IC50 = 2.6 nM T68547 C38DIF 134156853 IC50 = 180000 nM T68547 CI4W7T 134156856 IC50 = 12.8 nM T68547 C4FLQ5 134157355 IC50 > 100000 nM T68547 C1UP3S 134157845 IC50 = 2890 nM T68547 C9DSR3 134159676 IC50 = 21800 nM T68547 C0X1HQ 134224487 IC50 = 1270 nM T68547 CZV43J 134283792 IC50 = 15000 nM T68547 C62WXO 134283796 IC50 = 40000 nM T68547 CO7K3N 134283799 IC50 = 4400 nM T68547 CBQ17L 134283800 IC50 = 25000 nM T68547 C1Y4TA 134283810 IC50 = 35000 nM T68547 CV2YF7 134283813 IC50 = 29000 nM T68547 C05FVT 134492522 IC50 > 10000 nM T68547 CWJ7D1 134611695 IC50 = 2690 nM T68547 CE8IT7 134611723 Ki = 0.58 nM T68547 C1F6WZ 134812689 IC50 = 8 nM T68547 C7F0TV 134812690 IC50 > 1000000 nM T68547 CML7O0 134822021 IC50 = 21400 nM T68547 C52IBY 134823859 IC50 = 6900 nM T68547 C4Q6YP 135348847 IC50 > 30000 nM T68547 CU4F7J 135348851 IC50 > 30000 nM T68547 CYJ61T 135348854 IC50 = 11200 nM T68547 CJ1B8Z 135348856 IC50 > 30000 nM T68547 C14FWK 135348858 IC50 = 1390 nM T68547 CP90AW 135348876 IC50 > 30000 nM T68547 CJ9MO0 135348881 IC50 = 3030 nM T68547 CR1Z8J 135348908 IC50 > 30000 nM T68547 CS1V6A 135367138 IC50 > 50000 nM T68547 CVO59N 135367789 IC50 > 50000 nM T68547 CDY18W 135407493 IC50 > 100000 nM T68547 CW2I4R 135412048 IC50 > 100000 nM T68547 C7U0AV 135412194 IC50 > 100000 nM T68547 CI28ZH 135424818 IC50 = 572 nM T68547 CS54TL 135437514 IC50 = 82300 nM T68547 C36MUC 135441620 IC50 > 100000 nM T68547 CRB8M1 135444536 IC50 > 100000 nM T68547 CX5D6J 135446479 IC50 = 16400 nM T68547 C1TOK2 135449197 IC50 > 100000 nM T68547 CW25GL 135462117 IC50 > 100000 nM T68547 CCL28F 135473106 IC50 > 100000 nM T68547 CYA60G 135497781 IC50 > 100000 nM T68547 C01EZF 135567459 IC50 = 38000 nM T68547 CGB67N 135869606 IC50 = 200 nM T68547 CV3QP4 135886613 IC50 = 31.4 nM T68547 C8X5LO 135928012 Ki = 120 nM T68547 CI2YE8 135928628 IC50 > 100000 nM T68547 CWK65M 135981704 IC50 = 17 nM T68547 C5UXF8 135981705 IC50 = 18 nM T68547 C50NIS 136025837 IC50 > 100000 nM T68547 C4OS0V 136025842 IC50 > 100000 nM T68547 CX7Z5B 136025843 IC50 > 100000 nM T68547 CB8EM9 136025984 IC50 > 100000 nM T68547 C49MUG 136025986 IC50 > 100000 nM T68547 C0OLS8 136030779 IC50 = 41000 nM T68547 CIA7R4 136030780 IC50 > 100000 nM T68547 C24LKN 136030781 IC50 > 100000 nM T68547 CH7Y3C 136086920 IC50 > 100000 nM T68547 C3VDL5 136086921 IC50 > 100000 nM T68547 C9GOB5 136086922 IC50 = 77200 nM T68547 CE3ZL7 136086923 IC50 > 100000 nM T68547 CJZ5F3 136086924 IC50 > 100000 nM T68547 CT19ND 136110961 IC50 = 80 nM T68547 CY9U0E 136173089 IC50 = 100 nM T68547 C32MPU 136173094 IC50 = 100 nM T68547 CXHY69 136230092 IC50 = 1020 nM T68547 CWK9U7 136230093 IC50 = 660 nM T68547 C19VDS 136237971 IC50 = 839 nM T68547 CBS97C 136239447 IC50 = 930 nM T68547 CT2MI6 136239448 IC50 = 180 nM T68547 CE2F9G 136244081 IC50 = 370 nM T68547 C9CH7S 136244085 IC50 = 920 nM T68547 C5J2AX 136244086 IC50 = 410 nM T68547 CILG36 136286746 IC50 = 8 nM T68547 C39WRP 136286747 IC50 = 10500 nM T68547 C7ZX5O 136286761 IC50 = 673 nM T68547 C9SV6G 136645392 IC50 = 5860 nM T68547 CANQ56 136645396 IC50 = 937 nM T68547 C9TGH1 136645397 IC50 = 1810 nM T68547 C1F7JV 136645401 IC50 > 20000 nM T68547 C32LNQ 136645404 IC50 = 2030 nM T68547 C4W0IE 136645405 IC50 = 2880 nM T68547 CMIU28 136645406 IC50 = 9270 nM T68547 C3K2WL 136645410 IC50 = 1080 nM T68547 CC1D0X 136645415 IC50 = 7810 nM T68547 C02RIK 136645417 IC50 = 12900 nM T68547 C8CT0Z 136645422 IC50 = 357 nM T68547 CAWT82 136645431 IC50 = 335 nM T68547 CBZ8Q1 136645433 IC50 = 5980 nM T68547 C21EJD 136645435 IC50 = 490 nM T68547 C1KTV3 136645436 IC50 = 7200 nM T68547 CK1B9W 136645438 IC50 = 326 nM T68547 C6QOP7 136645441 IC50 = 387 nM T68547 CMZ71T 136645444 IC50 > 20000 nM T68547 CL47WS 136645445 IC50 = 276 nM T68547 C64BZR 136645447 IC50 = 7080 nM T68547 C7X1UL 136645449 IC50 = 286 nM T68547 CI9ZO7 136645454 IC50 = 1830 nM T68547 CA3I8S 136645455 IC50 = 4100 nM T68547 CRN16W 136645457 IC50 = 356 nM T68547 CGQ92L 136645458 IC50 = 1340 nM T68547 CO5DN2 136645462 IC50 = 1100 nM T68547 CRPN39 136645466 IC50 = 345 nM T68547 CL5X3G 136645467 IC50 = 2230 nM T68547 C48HNY 136959539 IC50 = 443 nM T68547 C1P8ZW 136959550 IC50 = 68 nM T68547 CKU95F 136966187 IC50 = 118 nM T68547 CFRG19 136985286 IC50 > 20000 nM T68547 CE7F4O 136985287 IC50 = 25 nM T68547 CFPT21 136985288 IC50 = 406 nM T68547 CBH5Y0 136985291 IC50 = 603 nM T68547 CDAK28 136985292 IC50 = 57 nM T68547 CQ9XW7 136985295 IC50 = 1530 nM T68547 C1M6NW 136985296 IC50 = 1110 nM T68547 CJOA28 136985302 IC50 = 793 nM T68547 CE6QK0 137125258 IC50 = 78 nM T68547 CAW80Q 137125259 IC50 = 200 nM T68547 C5CKZ8 137125261 IC50 = 82 nM T68547 C1ROQ9 137125262 IC50 = 130 nM T68547 CL29YN 137125263 IC50 = 530 nM T68547 C5OY8K 137125264 IC50 = 190 nM T68547 C0YGR6 137125265 IC50 = 240 nM T68547 CI78CK 137125267 IC50 = 290 nM T68547 CE8NM5 137125269 IC50 = 260 nM T68547 CANS59 137136982 IC50 > 20000 nM T68547 CDR9X0 137174935 IC50 = 150 nM T68547 CM1N3O 137226378 IC50 = 82250 nM T68547 C5AE3Q 137283418 IC50 > 20000 nM T68547 C5QIX1 137289788 IC50 = 554 nM T68547 C5X0YR 137289866 IC50 = 63 nM T68547 CU70ZB 137289868 IC50 = 7620 nM T68547 CV6AN7 137289892 IC50 > 20000 nM T68547 CB14CI 137289900 IC50 > 20000 nM T68547 CLY69S 137289946 IC50 = 2420 nM T68547 CC5HA4 137290225 IC50 > 20000 nM T68547 C4RBC7 137290234 IC50 = 2360 nM T68547 CKJ6Q4 137290238 IC50 = 4810 nM T68547 CR53GQ 137290273 IC50 = 225 nM T68547 C8DYG6 137290344 IC50 = 346 nM T68547 C9G3JB 137292402 IC50 = 14 nM T68547 C6MXL3 137292504 IC50 = 1880 nM T68547 CAZ49O 137300702 IC50 = 354 nM T68547 CGE0J6 137300703 IC50 = 3510 nM T68547 CDU43L 137300704 IC50 = 2440 nM T68547 CK0QG6 137300705 IC50 > 20000 nM T68547 C91IPL 137300706 IC50 = 6910 nM T68547 C5UYP8 137300707 IC50 = 6420 nM T68547 CHSG63 137300708 IC50 = 566 nM T68547 CX57MR 137300709 IC50 = 2610 nM T68547 C54KGS 137300710 IC50 = 66 nM T68547 CQD07Z 137300711 IC50 = 8750 nM T68547 C3I1CB 137300712 IC50 = 1530 nM T68547 C9LP2B 137353123 IC50 = 520 nM T68547 CNKJ27 137353141 IC50 = 1500 nM T68547 CAW4X1 137353146 IC50 = 760 nM T68547 CAPH58 137353182 IC50 = 2300 nM T68547 C4VXT3 137553162 IC50 = 86 nM T68547 CA5OY1 137628667 IC50 = 66.5 nM T68547 C67EFJ 137628684 IC50 = 0.19 nM T68547 CG23FD 137631444 IC50 = 9990 nM T68547 C9UQD2 137631509 IC50 > 30000 nM T68547 CP0JL9 137631552 IC50 > 30000 nM T68547 COL7W5 137631559 IC50 = 3.1 nM T68547 CHL7E8 137631592 IC50 = 58.8 nM T68547 CHYF09 137631675 IC50 = 620 nM T68547 CP0BN3 137631704 Ki > 50000 nM T68547 C31MPL 137631726 IC50 = 43.2 nM T68547 CJ9GD5 137631769 IC50 > 30000 nM T68547 CJ7P1U 137631803 IC50 = 49.6 nM T68547 CQ54WK 137631915 IC50 > 30000 nM T68547 CWSC97 137632010 IC50 = 0.84 nM T68547 CD1L0I 137632135 IC50 > 30000 nM T68547 C6A4GK 137632422 IC50 > 30000 nM T68547 CDLI15 137632451 IC50 = 39 nM T68547 CQ4BK9 137632561 IC50 > 30000 nM T68547 C28ZQV 137632620 IC50 = 433 nM T68547 CVB93K 137632723 IC50 = 12670 nM T68547 CW3PD2 137632740 IC50 = 260 nM T68547 C9RWF1 137632979 IC50 > 30000 nM T68547 CI2G7B 137633049 IC50 > 30000 nM T68547 CMU42D 137633092 IC50 > 30000 nM T68547 CY08AM 137633123 IC50 > 30000 nM T68547 C84MIY 137633138 IC50 = 48 nM T68547 CN1L0A 137633324 IC50 > 5000 nM T68547 CZY46A 137633389 IC50 = 10400 nM T68547 C1HL3I 137633415 IC50 > 30000 nM T68547 CS1LZ9 137633421 IC50 = 56.84 nM T68547 C37CRF 137633441 IC50 = 1.4 nM T68547 CM6V3G 137633491 IC50 = 99.91 nM T68547 C46IBX 137633497 IC50 = 19.21 nM T68547 CW8G1H 137633768 IC50 = 53.68 nM T68547 C82QCH 137633786 IC50 = 157.62 nM T68547 C5BZM4 137634010 IC50 = 4 nM T68547 C73PDL 137634086 IC50 = 24 nM T68547 C1V8QE 137634156 IC50 = 1000 nM T68547 C2OC5K 137634207 IC50 = 36 nM T68547 C8G4KJ 137634562 IC50 > 30000 nM T68547 CJ76DN 137634596 IC50 > 30000 nM T68547 C7JK8D 137634598 IC50 = 257.88 nM T68547 C7U1CE 137634604 IC50 > 30000 nM T68547 C6L3HN 137634634 IC50 = 2.2 nM T68547 C2ZLH6 137634772 IC50 = 250 nM T68547 C28CEY 137634881 IC50 = 75.12 nM T68547 C90TSR 137634950 IC50 > 30000 nM T68547 CZ1FK2 137635119 IC50 = 9.54 nM T68547 CS27YB 137635150 IC50 = 204 nM T68547 CHA4E3 137635225 IC50 = 13950 nM T68547 C6JVG9 137635398 IC50 = 6.9 nM T68547 CBMN61 137635405 IC50 > 30000 nM T68547 CAWZ25 137635575 IC50 = 1.34 nM T68547 CZ29MT 137635651 IC50 = 22870 nM T68547 COF8J3 137635708 IC50 = 29.9 nM T68547 C7N5BG 137635855 IC50 > 30000 nM T68547 CPL42O 137635914 IC50 = 84 nM T68547 C2KS3O 137635975 IC50 = 2700 nM T68547 C2MB4U 137636234 IC50 = 16840 nM T68547 CA2S3J 137636481 IC50 = 1440 nM T68547 C63ZFX 137636534 IC50 = 2650 nM T68547 C5GCO8 137636604 IC50 > 30000 nM T68547 CSY3E1 137636623 IC50 = 25000 nM T68547 C72SBN 137636632 IC50 > 30000 nM T68547 CQ4FP7 137636752 IC50 = 41 nM T68547 C9THE6 137636891 IC50 > 30000 nM T68547 CK1S0F 137637029 IC50 = 1.6 nM T68547 C8FH1S 137637247 IC50 = 138 nM T68547 CF3E8T 137637310 IC50 > 30000 nM T68547 C0VNM5 137637430 IC50 = 117.28 nM T68547 C7OT8F 137637596 IC50 = 300 nM T68547 C6MVX0 137637661 IC50 = 15700 nM T68547 C3H2GO 137637718 IC50 = 7990 nM T68547 CSH08B 137637787 IC50 > 30000 nM T68547 CEI0W2 137637915 IC50 = 2100 nM T68547 CZU9E2 137637958 IC50 = 29.81 nM T68547 CMU93I 137637990 IC50 > 30000 nM T68547 C6X0AW 137638091 IC50 = 45.02 nM T68547 CMD89K 137638151 IC50 = 11230 nM T68547 CQ3DR6 137638257 IC50 = 9000 nM T68547 CO9UY1 137638342 IC50 > 30000 nM T68547 C42PIU 137638406 IC50 = 300 nM T68547 C5FGB4 137638429 IC50 = 21 nM T68547 CF97LQ 137638432 IC50 > 5000 nM T68547 CW6F2I 137638447 IC50 = 25.66 nM T68547 C3RC2O 137638626 IC50 > 30000 nM T68547 C52GLN 137638676 IC50 = 798 nM T68547 CEMX30 137638687 IC50 > 30000 nM T68547 CTUL07 137638741 IC50 = 1.28 nM T68547 CP6NM0 137638747 IC50 = 93 nM T68547 CTG6X0 137638748 IC50 > 30000 nM T68547 CZP21J 137638798 IC50 > 5000 nM T68547 CDWG31 137638917 IC50 = 80.19 nM T68547 CZU31H 137638926 IC50 = 6180 nM T68547 CQ86FE 137638947 IC50 > 30000 nM T68547 C7IJC2 137639014 IC50 = 6430 nM T68547 C69IOZ 137639088 IC50 = 51.9 nM T68547 C0J8ZG 137639219 IC50 = 3540 nM T68547 CUG0C9 137639328 IC50 > 10000 nM T68547 C2DIM1 137639536 IC50 = 5270 nM T68547 CJBF37 137639551 IC50 = 129.57 nM T68547 CW4DJ8 137639563 IC50 > 30000 nM T68547 CS9A6C 137639566 IC50 > 30000 nM T68547 CMI6Z0 137639764 IC50 = 4570 nM T68547 C3CD6L 137639796 IC50 = 138.76 nM T68547 COV42L 137639829 IC50 > 30000 nM T68547 CL02GC 137640047 IC50 = 13880 nM T68547 C06BYV 137640258 IC50 = 28.88 nM T68547 CF7XJ2 137640263 IC50 = 440 nM T68547 C19GDO 137640291 IC50 = 17.5 nM T68547 CGKA54 137640295 IC50 > 30000 nM T68547 C7VIL6 137640304 IC50 = 22530 nM T68547 C3HRP7 137640379 IC50 = 500 nM T68547 C0Q3ZW 137640468 IC50 > 30000 nM T68547 C7HF0W 137640828 IC50 = 14500 nM T68547 CBQ7Z9 137640884 IC50 = 220 nM T68547 CIDW39 137640914 IC50 > 5000 nM T68547 CS50ET 137641009 IC50 = 1850 nM T68547 C39FQX 137641152 IC50 > 30000 nM T68547 CSA84O 137641263 IC50 = 4630 nM T68547 C3V4KQ 137641382 IC50 = 854 nM T68547 CI4PM3 137641395 IC50 > 30000 nM T68547 C4OEC3 137641520 IC50 = 1100 nM T68547 C5JUR2 137641533 IC50 = 627 nM T68547 C2G0XD 137641566 IC50 = 870 nM T68547 CS1K3I 137641616 IC50 > 30000 nM T68547 C38HXT 137641735 IC50 > 30000 nM T68547 CV19SL 137642038 IC50 > 30000 nM T68547 CF4X1L 137642042 IC50 > 5000 nM T68547 CTJA80 137642143 IC50 = 33 nM T68547 C7HKW1 137642159 IC50 = 72.27 nM T68547 CAF1N9 137642211 IC50 = 73.73 nM T68547 C48UDJ 137642293 IC50 = 903 nM T68547 C40JZA 137642448 IC50 > 30000 nM T68547 CKPB85 137642609 IC50 = 265 nM T68547 CY02GK 137642671 IC50 > 30000 nM T68547 C7MOD4 137642692 IC50 = 34.58 nM T68547 C1PRH5 137642860 IC50 = 24.7 nM T68547 C37BJQ 137642900 IC50 = 32.9 nM T68547 CQF49N 137643043 IC50 = 18700 nM T68547 CF42GI 137643288 IC50 = 143.25 nM T68547 C5QC2N 137643440 IC50 = 77.3 nM T68547 CJOS87 137643760 IC50 = 137 nM T68547 C4V1WC 137643841 IC50 = 9240 nM T68547 CB59SN 137643993 IC50 = 116.23 nM T68547 CWTP84 137644020 IC50 = 27 nM T68547 C7DLO4 137644089 IC50 = 55.5 nM T68547 CC38FN 137644424 IC50 > 30000 nM T68547 CVQ4J0 137644605 IC50 > 30000 nM T68547 CX37VS 137644658 IC50 > 30000 nM T68547 C1TKW9 137644960 IC50 = 3300 nM T68547 CCBN61 137645084 IC50 = 58.4 nM T68547 CTYM96 137645170 IC50 = 423 nM T68547 CPL3J1 137645258 IC50 > 30000 nM T68547 C8GNS5 137645287 IC50 = 467.82 nM T68547 C8XAR3 137645372 IC50 > 30000 nM T68547 C8WPM4 137645400 IC50 = 1600 nM T68547 CI8YV3 137645454 IC50 = 19100 nM T68547 C84JEV 137645469 IC50 = 330 nM T68547 CYA81D 137645509 IC50 = 71 nM T68547 C05LHW 137645511 IC50 > 30000 nM T68547 CX3E0H 137645675 IC50 = 20.6 nM T68547 C5REZ8 137645689 IC50 > 20000 nM T68547 CYSU67 137645967 IC50 > 30000 nM T68547 C8HKU4 137646033 IC50 = 137.85 nM T68547 CT98PM 137646118 IC50 = 100 nM T68547 CV7F6C 137646133 IC50 = 460 nM T68547 CMJ7D9 137646202 IC50 > 30000 nM T68547 CN08DL 137646214 IC50 > 30000 nM T68547 C6FPB8 137646630 IC50 = 83 nM T68547 C4K5JC 137646664 IC50 = 46 nM T68547 C3AIC9 137646743 IC50 = 370 nM T68547 CQI0Y6 137646988 IC50 = 1.6 nM T68547 CNT3Y7 137647005 IC50 = 246.57 nM T68547 C4I9YE 137647260 IC50 > 30000 nM T68547 CX8C9V 137647325 IC50 > 30000 nM T68547 CA0V2Q 137647353 IC50 = 96.4 nM T68547 CHW8X4 137647384 IC50 > 30000 nM T68547 CGMN16 137647616 Ki > 50000 nM T68547 CM65KH 137647813 IC50 = 1.06 nM T68547 C5AFM1 137647889 IC50 = 122.49 nM T68547 CZ2RN9 137647935 IC50 = 16920 nM T68547 CO7H5A 137648171 IC50 = 23 nM T68547 CI05DA 137648221 IC50 = 180 nM T68547 C5IK9F 137648357 IC50 = 174.73 nM T68547 C8S2TO 137648573 IC50 > 30000 nM T68547 C0VAB8 137648585 IC50 > 30000 nM T68547 CD9S6Y 137648608 IC50 = 37 nM T68547 CPK7Y5 137648623 IC50 > 30000 nM T68547 CL0XW1 137648762 IC50 = 3840 nM T68547 CR0P6Z 137648837 IC50 = 4550 nM T68547 CN3I9X 137648982 IC50 = 14.7 nM T68547 CG2PL8 137648996 IC50 = 17380 nM T68547 C05DNH 137649390 IC50 > 30000 nM T68547 CO20AE 137649565 IC50 > 30000 nM T68547 C7MHG2 137649586 IC50 = 7.18 nM T68547 C0PGD9 137649617 IC50 = 36.5 nM T68547 CGK2M9 137649620 IC50 = 40 nM T68547 CM15FY 137649624 IC50 = 6910 nM T68547 CDXE54 137649646 Ki > 50000 nM T68547 CE67ZS 137649860 IC50 > 30000 nM T68547 CH0ES8 137650022 IC50 > 30000 nM T68547 CRP0D7 137650200 IC50 = 11.27 nM T68547 C3AB2X 137650291 IC50 = 470 nM T68547 CQ5WF3 137650342 IC50 = 32 nM T68547 C7I9FA 137650637 IC50 = 2.6 nM T68547 C4MC5X 137650991 IC50 > 30000 nM T68547 C3VM4T 137651193 IC50 = 7.8 nM T68547 C4GNA5 137651338 IC50 > 30000 nM T68547 CEP9R0 137651700 IC50 = 1930 nM T68547 CA4FM3 137651729 IC50 = 72.5 nM T68547 C8PWX1 137651771 IC50 > 30000 nM T68547 CGE1Z5 137651786 IC50 > 30000 nM T68547 CD89ZR 137651966 IC50 > 30000 nM T68547 C3EQ0D 137651991 IC50 = 54.46 nM T68547 CT05IE 137651994 IC50 = 5900 nM T68547 CFLX25 137652000 IC50 = 2130 nM T68547 CH0TI5 137652048 IC50 = 912.5 nM T68547 CH3B5G 137652131 IC50 > 30000 nM T68547 C8NHK9 137652359 IC50 > 5000 nM T68547 C5FHD3 137652442 IC50 = 4320 nM T68547 CMP7G0 137652638 IC50 = 91.7 nM T68547 CB15PI 137652670 Ki > 50000 nM T68547 C83RBI 137652888 IC50 = 14970 nM T68547 CPI06O 137652951 IC50 = 54.27 nM T68547 CY73RL 137652969 IC50 > 5000 nM T68547 C7SUM3 137653261 IC50 = 220 nM T68547 CZI5S2 137653293 IC50 = 2740 nM T68547 C3QX5N 137653295 IC50 = 29.78 nM T68547 CE6UI4 137653337 IC50 > 5000 nM T68547 C61VOF 137653427 IC50 = 8510 nM T68547 COG3A4 137653572 IC50 = 29300 nM T68547 CQYF78 137653683 IC50 = 53 nM T68547 C82RZU 137653956 IC50 = 1600 nM T68547 CXZ5J3 137654094 IC50 = 27.4 nM T68547 C1OAE9 137654162 IC50 = 6540 nM T68547 C3FEM8 137654512 IC50 = 1510 nM T68547 C39QLZ 137654517 IC50 = 95 nM T68547 C1HE8S 137654622 IC50 = 27.26 nM T68547 CFQ4T2 137654668 IC50 > 30000 nM T68547 CTN10F 137654680 IC50 = 170 nM T68547 CCR5B3 137654793 IC50 = 6 nM T68547 C1SBN5 137654946 IC50 = 573.43 nM T68547 C9ONX3 137654984 IC50 = 0.53 nM T68547 C4OF1K 137655138 IC50 > 5000 nM T68547 CLWF87 137655165 IC50 > 30000 nM T68547 CV89YB 137655268 IC50 = 983 nM T68547 C79HAZ 137655524 IC50 = 350 nM T68547 CS50BH 137655597 IC50 > 30000 nM T68547 CN70IL 137655615 IC50 = 17 nM T68547 CZ5Y4F 137655761 IC50 = 3.8 nM T68547 C5EB0H 137655853 IC50 = 14.35 nM T68547 C2RKM4 137656021 IC50 = 180 nM T68547 C71ZNJ 137656226 IC50 = 5720 nM T68547 CIA0V1 137656228 IC50 > 30000 nM T68547 CQ23FB 137656234 IC50 = 3 nM T68547 CVG9T3 137656290 IC50 = 12 nM T68547 CI6R3W 137656303 Ki > 50000 nM T68547 C0NR1V 137656498 IC50 = 2010 nM T68547 CRP0T2 137656638 IC50 = 4010 nM T68547 CM7C0N 137656735 IC50 = 710 nM T68547 C9PUK8 137656850 IC50 = 670 nM T68547 C0EQI2 137656898 IC50 = 58.6 nM T68547 C76OGQ 137656942 IC50 = 8100 nM T68547 CY8A2I 137656945 IC50 = 95.46 nM T68547 C5BM7T 137657586 IC50 = 511 nM T68547 C97QUM 137657678 IC50 = 171 nM T68547 CR6B5H 137657803 IC50 = 14500 nM T68547 C21XDS 137657845 IC50 = 2900 nM T68547 C1DL3P 137657892 Ki > 50000 nM T68547 CYLD90 137658075 IC50 = 8.1 nM T68547 CN0C1E 137658519 IC50 > 30000 nM T68547 C8D2GT 137658785 Ki > 50000 nM T68547 CO5E2F 137658815 IC50 = 280 nM T68547 COC9D2 137658833 IC50 > 30000 nM T68547 CPJL30 137659007 IC50 = 284 nM T68547 CE49SB 137659150 IC50 = 100 nM T68547 C9D7NR 137659196 IC50 = 52.77 nM T68547 C1C8HZ 137659782 IC50 = 87 nM T68547 CFGW13 137659898 IC50 = 46 nM T68547 C6XWP9 137659968 IC50 = 141.12 nM T68547 CM0OE5 137660128 IC50 = 2250 nM T68547 CW5FQ4 137660152 IC50 = 28700 nM T68547 C6POG5 137660155 IC50 = 240 nM T68547 CLWU57 137660171 IC50 = 91.59 nM T68547 CU2SH5 137660339 IC50 > 5000 nM T68547 C7JGX8 137660397 IC50 = 53.8 nM T68547 C3Q7PX 137660404 IC50 = 10960 nM T68547 CAOG59 137660901 IC50 = 200 nM T68547 C02BSL 137661253 IC50 = 91.99 nM T68547 C5VR2U 137661620 IC50 = 110 nM T68547 C2RNY3 137661648 IC50 = 9.1 nM T68547 C4B9EG 137661742 IC50 > 30000 nM T68547 CO7Q1H 137661848 IC50 = 25600 nM T68547 CEJI95 137661885 IC50 = 26 nM T68547 CEF18M 137661927 IC50 > 5000 nM T68547 CNBS41 137661968 IC50 = 1.6 nM T68547 CQAY45 137662133 IC50 > 30000 nM T68547 CA51OM 137662221 IC50 = 12 nM T68547 CYZ43W 137662281 IC50 = 62.25 nM T68547 CM3UF7 137700779 IC50 > 10000 nM T68547 CAQ62X 137701235 Ki = 0.27 nM T68547 CVA12U 138377601 IC50 = 11160 nM T68547 CIWG23 138393067 IC50 = 590 nM T68547 C7EM3I 138393071 IC50 = 2190 nM T68547 C4NFS3 138393072 IC50 = 820 nM T68547 CA3C4O 138454792 IC50 = 1.4 nM T68547 CIT72O 139302883 IC50 = 3.57 nM T68547 CN1TH8 139302889 IC50 = 80.98 nM T68547 C0R1MD 139302991 IC50 = 40.92 nM T68547 C3GJQ8 139303021 IC50 = 19.87 nM T68547 CN73DV 139303049 IC50 = 279 nM T68547 CFAU90 139303050 IC50 = 38.25 nM T68547 CKQB30 139303051 IC50 = 16.52 nM T68547 CN2UH1 139303146 IC50 = 3.59 nM T68547 CE81VG 139303149 IC50 = 2.64 nM T68547 C9DJ3B 139303559 IC50 = 14.68 nM T68547 CN4M1E 139325532 IC50 = 1300 nM T68547 C9EBI4 139325820 IC50 > 10000 nM T68547 CP73QO 141504704 IC50 = 1460 nM T68547 CX7K2H 141514151 IC50 = 604.4 nM T68547 CLJ9H5 141514152 IC50 = 1429.5 nM T68547 CH9K7L 141733188 IC50 = 5080 nM T68547 C7XI0V 141764754 IC50 = 1.8 nM T68547 C3DCP2 142446438 IC50 = 2040 nM T68547 CO6C7N 142489312 IC50 = 1800 nM T68547 C7B3JK 142489313 IC50 = 2500 nM T68547 CGT08I 142489314 IC50 = 1200 nM T68547 CF7K4G 142489316 IC50 = 5500 nM T68547 CM6LR2 142489318 IC50 = 1500 nM T68547 C42DBC 142489319 IC50 = 370 nM T68547 CH5Y8E 142489322 IC50 = 1200 nM T68547 C5MN8W 142489323 IC50 = 1100 nM T68547 CFYC82 142489328 IC50 = 1200 nM T68547 C4DKW7 142489330 IC50 = 1300 nM T68547 CDS81U 142489335 IC50 = 300 nM T68547 CMY8W1 142489337 IC50 > 10000 nM T68547 CD5E9S 142489342 IC50 = 1400 nM T68547 C65LBI 142489344 IC50 = 3200 nM T68547 CX0E9B 142505968 IC50 = 5390 nM T68547 CBJC50 142505992 IC50 = 5846 nM T68547 C7N8LV 142506025 IC50 = 1575 nM T68547 CKBF56 142506033 IC50 = 429 nM T68547 CLND62 142506170 IC50 > 100000 nM T68547 CGNQ74 142506189 IC50 = 3925 nM T68547 C1T3IQ 142506210 IC50 = 388 nM T68547 CEGV67 142506220 IC50 = 8434 nM T68547 CP5HF8 142506225 IC50 = 67870 nM T68547 C1COW3 145948735 IC50 > 10000 nM T68547 CZ6D7U 145948737 IC50 > 10000 nM T68547 CL1T5W 145948741 IC50 > 10000 nM T68547 C1GMF5 145948743 IC50 = 23.9 nM T68547 CCEB28 145948752 IC50 = 4870 nM T68547 CTO5X4 145948791 IC50 = 201 nM T68547 CP98HY 145948798 IC50 > 10000 nM T68547 C43XJI 145948810 IC50 > 10000 nM T68547 C3JMP9 145948813 IC50 = 9910 nM T68547 C7K1WB 145948814 IC50 = 33.3 nM T68547 CFU6J8 145948816 IC50 > 10000 nM T68547 CG1Y3W 145948818 IC50 = 109 nM T68547 CAY43C 145948836 IC50 > 10000 nM T68547 CKI3Y2 145948841 IC50 = 68.6 nM T68547 C7JWF3 145948843 IC50 = 101 nM T68547 CJG3B6 145948850 IC50 = 652 nM T68547 CGKI09 145948851 IC50 = 613 nM T68547 CZ16SK 145948852 IC50 = 203 nM T68547 CA6W8I 145948853 IC50 > 10000 nM T68547 CF0Q3C 145948854 IC50 > 10000 nM T68547 CTEI37 145948871 IC50 = 533 nM T68547 C0VTX8 145948874 IC50 > 10000 nM T68547 C8FHP2 145948903 IC50 = 1650 nM T68547 C7RLZ8 145948904 IC50 > 10000 nM T68547 CE4WS8 145948905 IC50 = 16.1 nM T68547 C1KO6S 145948906 IC50 = 3690 nM T68547 C5EKH9 145948907 IC50 = 145 nM T68547 C5HL4D 145948914 IC50 = 531 nM T68547 C74UFN 145948956 IC50 = 79.5 nM T68547 CY09KL 145948957 IC50 = 160 nM T68547 CH91ER 145948958 IC50 = 2550 nM T68547 CE38KZ 145948959 IC50 = 316 nM T68547 CE15JW 145948961 IC50 = 923 nM T68547 CN6YM2 145948964 IC50 > 10000 nM T68547 CY49SE 145948983 IC50 > 10000 nM T68547 CH0UZ1 145948985 IC50 > 10000 nM T68547 C7Y5PK 145948986 IC50 = 50.4 nM T68547 CY1KB9 145949010 IC50 = 207 nM T68547 C1JMN9 145949196 IC50 = 980 nM T68547 C3M7JG 145949513 IC50 = 410 nM T68547 CDA28I 145949712 IC50 = 15 nM T68547 CXEV29 145949841 IC50 = 6070 nM T68547 CXJ0Y4 145949850 IC50 = 70 nM T68547 C1G2PB 145949937 IC50 = 3700 nM T68547 C1EF9X 145950102 IC50 = 27 nM T68547 CF54HP 145950469 IC50 = 310 nM T68547 C4W0YE 145950607 IC50 = 95 nM T68547 C9SMA8 145950715 IC50 = 100 nM T68547 CRKM19 145950884 IC50 = 2 nM T68547 CV3QO5 145951170 IC50 = 29.3 nM T68547 CMOW75 145951496 IC50 > 20000 nM T68547 CRSM78 145952088 IC50 > 160000 nM T68547 CMZ58R 145952121 IC50 = 3590 nM T68547 CFE4G6 145952135 IC50 = 58 nM T68547 CEC68O 145952295 IC50 = 1200 nM T68547 C4BZ0E 145952449 IC50 = 2900 nM T68547 CV5QI2 145952910 IC50 = 2920 nM T68547 CKG98W 145953085 IC50 > 20000 nM T68547 CA13YG 145953228 IC50 = 24000 nM T68547 C7I0VX 145953295 IC50 > 30000 nM T68547 CL0XT8 145954248 IC50 = 12 nM T68547 C4IC5P 145954578 IC50 = 380 nM T68547 CM53ZB 145954785 IC50 = 4120 nM T68547 CYD83K 145954811 IC50 = 910 nM T68547 CI62ZD 145955000 IC50 = 250 nM T68547 CNB9E6 145955015 IC50 = 610 nM T68547 C6QI4B 145955113 IC50 = 1700 nM T68547 C5FU6W 145955202 IC50 = 36 nM T68547 C23ZAQ 145955356 IC50 = 44 nM T68547 CGP9X1 145955496 IC50 = 38 nM T68547 CZ0K1H 145955759 IC50 = 2200 nM T68547 CW2VZ6 145955763 IC50 > 50000 nM T68547 CIK4T9 145955799 IC50 = 5100 nM T68547 CUM12F 145956028 IC50 = 9720 nM T68547 CM6UC8 145956323 IC50 = 1130 nM T68547 C7B2EU 145956761 IC50 = 46 nM T68547 C3XI4V 145956897 IC50 = 91 nM T68547 CBED35 145957183 IC50 = 4200 nM T68547 CFG58P 145957238 IC50 > 30000 nM T68547 CAP1Y3 145957299 IC50 = 890 nM T68547 CS6K8G 145957478 IC50 = 970 nM T68547 CJ03TU 145957740 IC50 = 218 nM T68547 CBNG29 145957781 IC50 = 38 nM T68547 C1R8DB 145957798 IC50 = 970 nM T68547 C9RH8U 145957804 IC50 = 2100 nM T68547 CJZ25F 145958256 IC50 = 3510 nM T68547 CMY49F 145958259 IC50 = 270 nM T68547 C5XP1C 145958407 IC50 = 350 nM T68547 C3L8IE 145958641 IC50 = 160 nM T68547 C8SI2G 145958925 IC50 > 10000 nM T68547 C18ZGV 145959245 IC50 = 60 nM T68547 C8RXN1 145959262 IC50 > 20000 nM T68547 CO05IK 145959360 IC50 = 18 nM T68547 CTPK43 145959386 IC50 = 890 nM T68547 CU78RJ 145959742 IC50 = 1010 nM T68547 C9IV1C 145959866 IC50 = 4.5 nM T68547 CFC18Z 145960569 IC50 = 1100 nM T68547 CK1XI0 145960971 IC50 > 10000 nM T68547 CAGS83 145961653 IC50 = 2700 nM T68547 C1X5EO 145962694 IC50 = 36 nM T68547 C29PAL 145963897 IC50 = 18000 nM T68547 CJ47DY 145964043 IC50 > 100000 nM T68547 C3PWD4 145964064 IC50 = 1440 nM T68547 CRO27A 145964093 IC50 > 1000 nM T68547 CEX67F 145964240 IC50 = 7300 nM T68547 CEDK05 145964533 IC50 = 1500 nM T68547 CDO47P 145964554 IC50 = 4400 nM T68547 CIME61 145964672 IC50 = 156 nM T68547 CDY56B 145964885 IC50 = 1460 nM T68547 CW6UM7 145965159 IC50 = 340 nM T68547 COH6A8 145965638 IC50 = 18 nM T68547 CZ9QK6 145965864 IC50 = 221 nM T68547 C68UOR 145966334 IC50 = 467 nM T68547 CM6KY1 145966543 IC50 = 37000 nM T68547 CJAE67 145966594 IC50 = 3120 nM T68547 C8O6RY 145966838 IC50 > 1000 nM T68547 CUD38A 145967089 IC50 = 770 nM T68547 C19POY 145967140 IC50 = 3790 nM T68547 C3AN8V 145967490 IC50 = 730 nM T68547 C93JKN 145967593 IC50 = 2021 nM T68547 CD82XB 145967610 IC50 = 430 nM T68547 CT9W7K 145967676 IC50 = 1200 nM T68547 C7OG1D 145967698 IC50 = 1071 nM T68547 C0GY3Q 145967784 IC50 = 329 nM T68547 C5RPQ9 145967832 IC50 = 110 nM T68547 CI1ZD2 145967851 IC50 > 5000 nM T68547 COT40H 145967888 IC50 = 2800 nM T68547 CR59HK 145967905 IC50 = 1039 nM T68547 C95SNQ 145967968 IC50 = 836 nM T68547 CX0OD9 145968046 IC50 = 22.9 nM T68547 CES7W6 145968087 IC50 = 3611 nM T68547 C3LH2I 145968221 IC50 > 1000 nM T68547 CSO4I7 145968364 IC50 > 5000 nM T68547 C2XS8E 145968675 IC50 = 219 nM T68547 CSJ81Y 145968726 IC50 = 230 nM T68547 CG0S9U 145968824 IC50 = 1883 nM T68547 CIA79M 145968985 IC50 = 480 nM T68547 CH9JR8 145969001 IC50 = 900 nM T68547 C27YHM 145969456 IC50 = 79 nM T68547 CV53YN 145969651 IC50 = 487 nM T68547 C8RO9H 145969692 IC50 = 2500 nM T68547 C0K6XS 145969789 IC50 = 694 nM T68547 CUI37A 145969799 IC50 = 45.3 nM T68547 CWU27Z 145969804 IC50 = 2470 nM T68547 CZ80EP 145969996 IC50 = 925 nM T68547 C5ZB0M 145970020 IC50 = 1100 nM T68547 CME7W2 145970049 IC50 > 1000 nM T68547 C79YOL 145970069 IC50 = 27000 nM T68547 C7TSV2 145970161 IC50 = 3741 nM T68547 CG5OK8 145970171 IC50 = 66 nM T68547 C8FXH4 145970309 IC50 = 24000 nM T68547 CBR60K 145970453 IC50 = 541 nM T68547 C0E2UO 145970598 IC50 = 38 nM T68547 CI43DY 145970786 IC50 = 1320 nM T68547 C63KEL 145970838 IC50 > 100000 nM T68547 C7UG3O 145971121 IC50 > 100000 nM T68547 C7VD9I 145971506 IC50 = 2913 nM T68547 C4EU5J 145971645 IC50 > 1000 nM T68547 C7K1AJ 145971681 IC50 = 250 nM T68547 CZ85FJ 145972657 IC50 = 9200 nM T68547 CW0T7A 145973234 IC50 = 3480 nM T68547 CO51JK 145973368 IC50 = 36.2 nM T68547 C4HTO2 145973543 IC50 = 877 nM T68547 CFP2R3 145973876 IC50 = 18000 nM T68547 CVM0Z3 145974125 IC50 = 7160 nM T68547 CLCU89 145974270 IC50 = 1800 nM T68547 C8YEJ9 145974425 IC50 = 3300 nM T68547 CUJE21 145974558 IC50 > 10000 nM T68547 CY1G2F 145974565 IC50 = 314 nM T68547 C5YJO8 145974667 IC50 = 14000 nM T68547 C2NP6U 145975596 IC50 = 38 nM T68547 CE8I5V 145975869 IC50 = 1210 nM T68547 C6Y9QH 145975913 IC50 = 13000 nM T68547 C7ANI4 145976192 IC50 = 78 nM T68547 C86GXV 145976671 IC50 = 2400 nM T68547 CMUA94 145976675 IC50 = 1420 nM T68547 C8Z2IP 145976817 IC50 = 216 nM T68547 CN6UO4 145977003 IC50 = 8540 nM T68547 CKAQ67 145977127 IC50 = 2800 nM T68547 CSC6A1 145977313 IC50 = 129 nM T68547 C78XNS 145977336 IC50 = 57000 nM T68547 C8DBK1 145977522 IC50 > 1000 nM T68547 CLY4Z5 145977632 IC50 = 270 nM T68547 CCD9U2 145977675 IC50 = 625 nM T68547 CP53JS 145977717 IC50 = 3.9 nM T68547 C3QYB8 145978561 IC50 > 100000 nM T68547 CR1ZY6 145978627 IC50 > 1000 nM T68547 COR40V 145978805 IC50 = 4780 nM T68547 C7X4LZ 145978932 IC50 = 1380 nM T68547 CG4M5X 145979054 IC50 = 70.5 nM T68547 C91TLI 145979056 IC50 = 177 nM T68547 C7TAL5 145979161 IC50 = 3.8 nM T68547 C5SK4O 145979193 IC50 = 23.5 nM T68547 CFJ1L2 145979358 IC50 = 9.3 nM T68547 CCV92M 145979587 IC50 = 40 nM T68547 CFT50A 145979673 IC50 = 637 nM T68547 CZ7IQ9 145979841 IC50 = 4.7 nM T68547 CS3HT7 145979964 IC50 = 41 nM T68547 C0UG8S 145980171 IC50 = 1040 nM T68547 CZMP56 145980566 IC50 = 11440 nM T68547 CIM41N 145980574 IC50 = 253 nM T68547 CWH40Y 145980630 IC50 = 289 nM T68547 CX94BD 145980658 IC50 = 32.4 nM T68547 C09BPI 145980773 IC50 = 260 nM T68547 C9ZT8Y 145981096 IC50 = 3350 nM T68547 COG0N1 145981347 IC50 > 10000 nM T68547 CFR1P8 145981954 IC50 = 552 nM T68547 CMB08D 145981960 IC50 = 2490 nM T68547 C2OC6Q 145982084 IC50 = 1043 nM T68547 C9VDE5 145982499 IC50 = 440 nM T68547 CKYP15 145982514 IC50 = 12620 nM T68547 CF8R6Z 145982577 IC50 = 2 nM T68547 CX2LY1 145982614 IC50 = 5570 nM T68547 CHI03D 145982623 IC50 = 83 nM T68547 C2PFB5 145982658 Ki = 0.51 nM T68547 C6QGM5 145982769 IC50 = 3.9 nM T68547 C0SHF9 145982778 IC50 = 13620 nM T68547 C71AZC 145982856 IC50 = 1319 nM T68547 CN4T7U 145982897 IC50 = 63 nM T68547 C0Z6NV 145982900 Ki = 0.097 nM T68547 CA7K6C 145983002 IC50 = 1721 nM T68547 CWN68A 145983070 Ki = 2.5 nM T68547 C5TH0E 145983101 Ki = 0.15 nM T68547 CE5WL7 145983126 Ki = 7.3 nM T68547 CR63YW 145983218 IC50 = 110 nM T68547 CLY2K6 145983228 Ki = 1.9 nM T68547 C6OL1K 145983267 IC50 = 2990 nM T68547 CA1LM5 145983443 IC50 = 179 nM T68547 CPUJ75 145983482 IC50 = 11010 nM T68547 CXF9G4 145983559 IC50 = 306.2 nM T68547 C0SH7K 145983585 Ki = 0.69 nM T68547 CH9L5S 145983605 Ki = 0.39 nM T68547 CMY73B 145983639 IC50 = 2700 nM T68547 CWD0A9 145983712 Ki = 0.075 nM T68547 CBIL37 145983726 Ki = 0.057 nM T68547 C5UY0O 145983746 Ki = 0.28 nM T68547 C2I7EQ 145983818 IC50 = 19670 nM T68547 C34ZQV 145983855 IC50 = 133.8 nM T68547 CV8H2B 145983876 IC50 = 30090 nM T68547 C6UZO1 145983877 Ki = 0.056 nM T68547 C3I6VL 145983950 IC50 = 710 nM T68547 CJLG54 145984020 IC50 = 44 nM T68547 C7FBZ5 145984102 IC50 = 27660 nM T68547 C62UNC 145984122 IC50 = 14.1 nM T68547 CGW04D 145984128 Ki = 4.8 nM T68547 C8VP6L 145984237 Ki = 0.23 nM T68547 CL43AD 145984253 IC50 = 45 nM T68547 CE40NU 145984280 Ki = 11 nM T68547 CIWO70 145984314 IC50 = 1950 nM T68547 CODK63 145984420 IC50 = 101 nM T68547 C85CVL 145984470 Ki = 12 nM T68547 CMWV73 145984487 Ki = 12 nM T68547 C9ZKC1 145984665 IC50 = 2030 nM T68547 CX36SR 145984704 IC50 = 5.1 nM T68547 CM27PO 145984713 Ki = 2.3 nM T68547 C01OFR 145984762 Ki = 0.5 nM T68547 C6XP8Y 145984765 Ki = 4.3 nM T68547 CQR2L8 145984786 Ki = 2.3 nM T68547 CXWS04 145984852 IC50 = 2706 nM T68547 C5U2QK 145984896 IC50 = 308.1 nM T68547 CSA1K8 145984949 IC50 = 27090 nM T68547 CTX1H9 145984993 Ki = 9.4 nM T68547 C2ND4F 145985023 IC50 = 1997 nM T68547 CX8MU4 145985048 Ki = 0.56 nM T68547 CJF71C 145985091 IC50 = 66.2 nM T68547 CT50ZG 145985100 IC50 = 1960 nM T68547 C3KU4L 145985106 Ki = 11 nM T68547 CFLH65 145985111 IC50 = 17400 nM T68547 CCRK43 145985194 Ki = 0.063 nM T68547 CRO4V1 145985225 Ki = 2.7 nM T68547 CN6KB9 145985243 IC50 = 130 nM T68547 CT2O9Q 145985360 Ki = 0.27 nM T68547 CB24HO 145985400 IC50 = 480 nM T68547 C60TZP 145985422 IC50 = 8.2 nM T68547 CPN23X 145985485 Ki = 0.91 nM T68547 CVB45P 145985612 Ki = 0.29 nM T68547 CDM0T5 145985755 IC50 = 224.3 nM T68547 C1GLM7 145985897 Ki = 4.4 nM T68547 CK90XR 145985933 IC50 = 90 nM T68547 CBF13W 145985947 IC50 = 6180 nM T68547 CZ4JB1 145986013 Ki = 0.27 nM T68547 CWJ56L 145986183 Ki = 1.4 nM T68547 C56MWZ 145986208 Ki = 3.8 nM T68547 CL62QV 145986214 IC50 = 4450 nM T68547 CGN02Q 145986264 IC50 = 970 nM T68547 C51BUM 145986322 IC50 = 2.8 nM T68547 C3QCS5 145986385 IC50 = 121.1 nM T68547 C1WH7V 145986586 IC50 > 5000 nM T68547 CS79CE 145986632 IC50 = 150 nM T68547 C7L1GU 145986811 IC50 = 54.7 nM T68547 CFWH51 145987165 IC50 = 4000 nM T68547 CRSN59 145987267 IC50 = 590 nM T68547 C2XPR7 145987380 IC50 = 1701 nM T68547 CRX8H1 145987492 IC50 = 133 nM T68547 CFH27G 145987566 IC50 = 774 nM T68547 CPAX89 145987732 IC50 = 24 nM T68547 CJ1M7T 145987832 IC50 = 1.9 nM T68547 CR4YX8 145987935 IC50 = 428 nM T68547 CK6U7Z 145988024 IC50 = 89 nM T68547 CV3S8R 145988041 IC50 = 2570 nM T68547 C8XBL4 145988088 IC50 = 77 nM T68547 C3F6SR 145988345 IC50 = 632.7 nM T68547 CFRN35 145988434 IC50 = 46.2 nM T68547 CPT93U 145988661 IC50 = 8.2 nM T68547 C82CIN 145988785 IC50 > 30000 nM T68547 C0NI8A 145988806 IC50 = 139 nM T68547 C2EXQ1 145989123 IC50 = 4470 nM T68547 CJ9G5A 145989228 IC50 = 65 nM T68547 CI97FM 145989333 IC50 = 4581 nM T68547 CJ8DO3 145989487 IC50 = 352 nM T68547 CPHG80 145989625 IC50 = 219 nM T68547 CLK52R 145990092 IC50 = 9.2 nM T68547 C5UZ4J 145990125 IC50 = 304 nM T68547 CHR0U9 145990400 IC50 = 7.1 nM T68547 C4PSZ2 145990543 IC50 = 6790 nM T68547 CO7F1K 145990990 IC50 = 145 nM T68547 CKU2L4 145991209 IC50 = 47.7 nM T68547 CZ94XS 145991731 IC50 = 934 nM T68547 C6WN7O 145992050 IC50 = 11710 nM T68547 CQ90ZB 145992461 IC50 = 66.5 nM T68547 CJC47L 145992551 IC50 = 142 nM T68547 C3RC5J 145992581 IC50 = 384 nM T68547 C4CEN6 145992608 IC50 = 262.4 nM T68547 C84YXW 145992837 IC50 = 71 nM T68547 CD09RT 145992905 IC50 = 56 nM T68547 C68VKC 145993051 IC50 = 1020 nM T68547 C7I5XM 145993519 IC50 = 7290 nM T68547 C51ZNC 145993585 IC50 = 155 nM T68547 CF54BR 145993638 IC50 = 10870 nM T68547 CF36GI 145993689 IC50 = 348 nM T68547 C1W6CF 145994016 IC50 = 11000 nM T68547 CVL35T 145994129 IC50 = 894.8 nM T68547 CSQ7G0 145994254 IC50 = 83 nM T68547 C0GMR1 146585718 IC50 = 6067 nM T68547 CJYD03 146836277 IC50 = 1132 nM T68547 CF2YV5 147185900 IC50 = 558.1 nM T68547 C0YXS8 147254231 IC50 = 910 nM T68547 C3RB5F 147731349 IC50 = 259.6 nM T68547 CA1EC6 147746059 IC50 = 119.7 nM T68547 CV9M5L 147777638 IC50 = 1060 nM T68547 C7L2GO 147878620 IC50 = 5432 nM T68547 CKEG86 148044361 IC50 = 296.2 nM T68547 CBG8T7 148123770 IC50 = 98.02 nM T68547 C5KHE1 148150539 IC50 = 90.05 nM T68547 C48EXH 148289288 IC50 = 6.31 nM T68547 C3SA6B 148608442 IC50 = 15.2 nM T68547 CT5E1O 148634364 IC50 = 164.6 nM T68547 CWLF12 148743859 IC50 = 278.3 nM T68547 CWCP30 148853853 IC50 = 15707 nM T68547 COH3I8 148951442 IC50 = 83.71 nM T68547 CO47EC 148970856 IC50 = 36.3 nM T68547 C3EFX4 149016806 IC50 = 103 nM T68547 CN71OS 149405396 IC50 = 3069 nM T68547 CV5ZR0 149819902 IC50 = 9540 nM T68547 CH3JE4 150054712 IC50 = 10810 nM T68547 C8S3MF 150076000 IC50 > 300 nM T68547 C8BM2K 150127738 IC50 = 394.5 nM T68547 C9L7DG 150259632 IC50 = 18860 nM T68547 CKMU94 150304623 IC50 = 335.6 nM T68547 CU2XY0 150312795 IC50 = 14500 nM T68547 C5PQI9 150470306 IC50 = 11150 nM T68547 C4JP7X 150533939 IC50 = 8275 nM T68547 CAQ36F 150619353 IC50 = 12700 nM T68547 C89BKD 150622000 IC50 > 10000 nM T68547 C5T1PC 150863979 IC50 = 19101 nM T68547 CIM06Z 150916115 IC50 = 8021 nM T68547 CN46CZ 150945374 IC50 = 15915 nM T68547 CM6IF7 151532669 IC50 = 9080 nM T68547 CS0V6U 151543423 IC50 = 13410 nM T68547 CV39LB 151825687 IC50 > 10000 nM T68547 CA21YZ 151887635 IC50 = 12000 nM T68547 CF7NB5 151976649 IC50 = 79.81 nM T68547 CROU95 152148008 IC50 = 6655 nM T68547 CY1NG0 152157103 IC50 = 10870 nM T68547 CYF2I5 152375216 IC50 = 22940 nM T68547 CL1UA7 152547478 IC50 = 9410 nM T68547 C2AOQ6 152562172 IC50 = 13170 nM T68547 CP6YK7 153056786 IC50 = 470.1 nM T68547 CT4GI5 153155940 IC50 = 489 nM T68547 C4F8LC 153265113 IC50 = 291.6 nM T68547 C17DHQ 153406869 IC50 = 141.4 nM T68547 CA17JT 153406872 IC50 = 1158 nM T68547 CC35YT 153406873 IC50 = 118.4 nM T68547 C0VF5H 153406878 IC50 = 25486 nM T68547 CT4H9P 153408403 IC50 = 10430 nM T68547 CK7P3F 153408410 IC50 = 7374 nM T68547 C9FIY4 153534005 IC50 = 46 nM T68547 C7F1UK 155454897 IC50 = 3340 nM T68547 C6ISA2 155510865 IC50 = 42 nM T68547 CIG6K4 155510915 IC50 = 200 nM T68547 C1ZXV2 155511261 IC50 = 6.3 nM T68547 C0KW3O 155511274 IC50 = 56.32 nM T68547 CB8RS9 155512087 IC50 > 25000 nM T68547 C5K6RO 155512136 IC50 = 980 nM T68547 C7FO1Y 155512340 IC50 = 3.3 nM T68547 CV2MG0 155512401 IC50 = 34 nM T68547 C6ERK4 155512456 IC50 = 81 nM T68547 CT4VS3 155512474 IC50 = 33 nM T68547 CQ5BL7 155512551 IC50 > 50000 nM T68547 CGN9Y6 155512914 IC50 = 233 nM T68547 CIC87K 155512972 IC50 = 0.15 nM T68547 C7VKU2 155513116 IC50 = 20 nM T68547 CHLO32 155513171 IC50 = 1200 nM T68547 CJ8IQ0 155513281 IC50 = 4.9 nM T68547 CE4H7I 155513471 IC50 > 50000 nM T68547 CN9JW5 155513555 IC50 > 1000 nM T68547 CJ2WH6 155514239 IC50 = 70.3 nM T68547 CCDH73 155514314 IC50 = 3000 nM T68547 C6BV9W 155514532 IC50 = 1580 nM T68547 CW3VT9 155514603 IC50 > 50000 nM T68547 CXVL19 155514838 IC50 = 2.2 nM T68547 CZ84WI 155515284 IC50 > 50000 nM T68547 CWEZ05 155515488 IC50 = 0.46 nM T68547 CUKG21 155515602 IC50 > 50000 nM T68547 CR1JH7 155515739 IC50 > 1000 nM T68547 CW7Q1N 155515767 IC50 = 96.8 nM T68547 CY2DC1 155515836 IC50 = 27 nM T68547 CYJ53T 155515864 IC50 = 12000 nM T68547 C1K2XN 155516139 IC50 = 1674 nM T68547 CFD72J 155516184 IC50 = 3.7 nM T68547 CL47DJ 155516579 IC50 = 3750 nM T68547 CT7R5L 155516928 IC50 = 65.6 nM T68547 CNP25D 155516982 IC50 = 1.7 nM T68547 CA1J3N 155517086 IC50 = 194 nM T68547 CL72ME 155517175 IC50 = 1.23 nM T68547 C7G0XM 155517418 IC50 = 484 nM T68547 C7SEB5 155517457 IC50 = 303 nM T68547 CYS75R 155517555 IC50 = 1030 nM T68547 CVI9Y7 155517723 IC50 = 3990 nM T68547 CY54TU 155518062 IC50 = 12000 nM T68547 CEH2N5 155518106 IC50 = 959 nM T68547 CE7QS8 155518248 IC50 = 16610 nM T68547 C58ZNC 155518327 IC50 = 2.9 nM T68547 CCDU61 155518496 IC50 = 16 nM T68547 CAD06U 155519254 IC50 = 200 nM T68547 C8XCP4 155519431 IC50 = 3 nM T68547 CDY5H6 155519645 IC50 = 6060 nM T68547 C81SOG 155520064 IC50 = 2.5 nM T68547 C3MX5D 155520119 IC50 = 12000 nM T68547 C4P1RM 155520291 IC50 = 12780 nM T68547 C34FXY 155520399 IC50 = 2880 nM T68547 CS8F6V 155520526 IC50 = 57.9 nM T68547 CAD10S 155520741 IC50 > 10000 nM T68547 C4A1SF 155520751 IC50 = 491 nM T68547 CAZ3S7 155521187 IC50 = 8800 nM T68547 CAS23O 155521203 IC50 = 57 nM T68547 C30DXG 155521234 IC50 = 12.1 nM T68547 CZ75FW 155521272 IC50 = 111 nM T68547 CG4F2U 155521283 IC50 = 71 nM T68547 CR7K5H 155521373 IC50 = 19573 nM T68547 CSI2W0 155521586 IC50 = 13 nM T68547 CCV14N 155521717 IC50 = 5760 nM T68547 C82PHV 155521822 IC50 = 1980 nM T68547 C6DVZ9 155521965 IC50 = 1100 nM T68547 C0KJ1Z 155522601 IC50 = 8599 nM T68547 C9FNJ8 155523062 IC50 = 4 nM T68547 CP67LK 155523130 IC50 = 11.4 nM T68547 CEQ58R 155523224 IC50 = 5.2 nM T68547 CG84WO 155523907 IC50 = 610 nM T68547 CU5RZ1 155524034 IC50 = 168 nM T68547 CJ3E4G 155524660 IC50 = 5550 nM T68547 CB0GT4 155524669 IC50 = 52 nM T68547 CBP78G 155524778 IC50 = 774.7 nM T68547 CNW0D1 155524821 IC50 = 1.8 nM T68547 CX6QF0 155524910 IC50 = 27.5 nM T68547 CYK1M8 155524976 IC50 = 1.3 nM T68547 C23QFM 155525013 IC50 = 6 nM T68547 CI24AD 155525662 IC50 = 1089 nM T68547 CN7B1T 155525782 IC50 = 255 nM T68547 C31XHG 155526170 IC50 = 2.4 nM T68547 CG1K0O 155526247 IC50 = 9842 nM T68547 COD92I 155526258 IC50 = 915 nM T68547 C46UIC 155526269 IC50 = 2790 nM T68547 CV8J0O 155526623 IC50 = 43 nM T68547 C63NOC 155527045 IC50 = 221 nM T68547 CBQ8C5 155527116 IC50 = 122 nM T68547 CC9W3J 155527176 IC50 = 4.9 nM T68547 C9PI3H 155527271 IC50 = 5.3 nM T68547 CEM0A3 155527290 IC50 = 209.7 nM T68547 CW2H5R 155527295 IC50 = 62 nM T68547 CQK19H 155527955 IC50 = 103 nM T68547 COMJ49 155528093 IC50 = 9.7 nM T68547 C7SPF3 155528334 IC50 = 128.4 nM T68547 CF6NT5 155528400 IC50 = 29 nM T68547 CHR4K5 155528532 IC50 > 100000 nM T68547 CQ4RG3 155528629 IC50 = 3060 nM T68547 C0IC6W 155528706 IC50 = 1.3 nM T68547 CK67EB 155529012 IC50 = 3370 nM T68547 CZ70PO 155529066 IC50 > 50000 nM T68547 C49NGT 155529137 IC50 > 50000 nM T68547 C9L6OC 155529247 IC50 = 1.3 nM T68547 CX2OS7 155529270 IC50 = 7500 nM T68547 C70MEU 155529500 IC50 = 2.6 nM T68547 C95YJA 155529506 IC50 = 316.2 nM T68547 C94BFW 155529690 IC50 = 5460 nM T68547 C3ENZ5 155529741 IC50 = 466 nM T68547 CR3XJ8 155529775 IC50 = 350 nM T68547 C74OTA 155529983 IC50 = 620 nM T68547 CU0C7W 155530254 IC50 = 1000 nM T68547 CTQ2P0 155530465 IC50 = 2 nM T68547 CAKD69 155530558 IC50 = 197 nM T68547 CZMC49 155530597 IC50 = 2.5 nM T68547 C8AZI6 155530932 IC50 = 381.5 nM T68547 C47WTL 155531016 IC50 = 630 nM T68547 CZG79N 155531159 IC50 = 93.05 nM T68547 C0HAD6 155531290 IC50 = 8.2 nM T68547 C7U8YQ 155531296 IC50 = 8.9 nM T68547 CN3W5J 155531452 IC50 > 50000 nM T68547 CE7Q6O 155531509 IC50 = 37 nM T68547 CUC3P1 155531533 IC50 = 1160 nM T68547 CC0WN1 155531780 IC50 = 6190 nM T68547 CJ04LR 155531942 IC50 = 178 nM T68547 CK2UY4 155531957 IC50 > 50000 nM T68547 C02GPA 155531979 IC50 = 10 nM T68547 CDJ0W3 155532052 IC50 = 636 nM T68547 CZO38U 155532084 IC50 = 1262 nM T68547 C3HDI1 155532640 IC50 = 11.92 nM T68547 CD8ZV7 155532950 IC50 = 1030 nM T68547 CR0YB5 155533057 IC50 = 2.3 nM T68547 CIZ46A 155533876 IC50 = 4900 nM T68547 C0T8AS 155533910 IC50 = 381 nM T68547 CF69UC 155534005 IC50 = 1000 nM T68547 CK6W2Y 155534018 IC50 = 665 nM T68547 CPE68B 155534222 IC50 = 1258.93 nM T68547 CMXD31 155534843 IC50 = 161 nM T68547 CCGS79 155535013 IC50 = 166 nM T68547 C6LB5D 155535084 IC50 > 30000 nM T68547 C6O8JB 155535273 IC50 = 11 nM T68547 CF37GO 155535511 IC50 = 1620 nM T68547 CRI36G 155535653 IC50 = 9.3 nM T68547 CD49QF 155535974 IC50 = 7490 nM T68547 CO91WP 155536301 IC50 = 6810 nM T68547 CPTA48 155536355 IC50 = 320 nM T68547 CI3NY7 155536462 IC50 = 75 nM T68547 CH27XY 155536857 IC50 = 2080 nM T68547 C81KIF 155537008 IC50 = 10 nM T68547 C2JH0S 155537112 IC50 = 38 nM T68547 CX9EO1 155537184 IC50 = 11 nM T68547 C5A2WC 155537194 IC50 = 1.3 nM T68547 CYE06Z 155537200 IC50 = 4930 nM T68547 CQV6H0 155537405 IC50 = 2925 nM T68547 C5FRG0 155537455 IC50 = 58.12 nM T68547 CTF98X 155537473 IC50 = 590 nM T68547 CAG9P4 155537573 IC50 > 50000 nM T68547 CNO90C 155537865 IC50 = 20 nM T68547 CJ86WN 155538082 IC50 = 14.7 nM T68547 CTU3X6 155538087 IC50 = 1700 nM T68547 C50EMD 155538313 IC50 > 1000 nM T68547 C54PWX 155538438 IC50 = 7 nM T68547 C63FKN 155538445 IC50 = 430 nM T68547 CJ6SF9 155538658 IC50 = 7650 nM T68547 COWZ49 155538705 IC50 = 24 nM T68547 C1PFV7 155538765 IC50 = 385 nM T68547 CLD19W 155539311 IC50 = 1310 nM T68547 CU6V4Q 155539319 IC50 > 50000 nM T68547 CM5UN4 155539714 IC50 = 412.8 nM T68547 CE6G4A 155539837 IC50 = 22.33 nM T68547 CBO78Z 155540097 IC50 = 602 nM T68547 C6U0FM 155540189 IC50 = 24000 nM T68547 CH0J8Z 155540388 IC50 = 1860 nM T68547 C6LQT1 155540719 IC50 = 2524 nM T68547 CZ8OB3 155540741 IC50 = 65 nM T68547 CBC5O0 155541221 IC50 = 93 nM T68547 CKN07B 155541358 IC50 = 837 nM T68547 C7B5NU 155541992 IC50 = 6560 nM T68547 C4T9YC 155542195 IC50 > 100000 nM T68547 C5OQ3G 155542658 IC50 = 1.6 nM T68547 CN7E6U 155542755 IC50 = 300 nM T68547 C2D1OT 155542789 IC50 = 26 nM T68547 C13NSL 155542830 IC50 = 758 nM T68547 CJ25HV 155542887 IC50 = 12.9 nM T68547 CKH3C6 155543263 IC50 = 1600 nM T68547 CV2G1W 155544267 IC50 = 39 nM T68547 CP4L1F 155544459 IC50 = 38000 nM T68547 CPIQ21 155544472 IC50 = 16.1 nM T68547 CJK31W 155544599 IC50 = 2380 nM T68547 CNM3P1 155544603 IC50 > 10000 nM T68547 CXR86J 155545078 IC50 > 50000 nM T68547 CCV9J0 155545380 IC50 = 4.4 nM T68547 C7YOP9 155545823 IC50 = 996 nM T68547 C8DQ7U 155546022 IC50 = 29.43 nM T68547 C2E5RQ 155546107 IC50 = 2950 nM T68547 CE1D7Q 155546207 IC50 > 100000 nM T68547 CF2O4J 155546325 IC50 > 50000 nM T68547 CK45LA 155546486 IC50 = 1584.89 nM T68547 C3HB0U 155546555 IC50 = 316.23 nM T68547 CS3GO2 155546558 IC50 = 1980 nM T68547 C0AU1L 155546632 IC50 > 50000 nM T68547 C8LT4A 155546691 IC50 = 15.8 nM T68547 C7N5XC 155546755 IC50 = 50 nM T68547 CEF69A 155546817 IC50 = 5.6 nM T68547 CP3Q7I 155547009 IC50 = 4200 nM T68547 CHD0I6 155547367 IC50 = 596 nM T68547 CIQ8G6 155547573 IC50 = 2.1 nM T68547 CTFU61 155549051 IC50 = 380 nM T68547 C90FBZ 155549087 IC50 > 50000 nM T68547 CE0YL6 155549538 IC50 = 3200 nM T68547 CFA01C 155549905 IC50 = 163.4 nM T68547 CD37YN 155550342 IC50 = 61 nM T68547 CO2TF8 155550660 IC50 = 5.8 nM T68547 C8US1B 155550805 IC50 = 41.9 nM T68547 C4Z5JX 155550827 IC50 > 50000 nM T68547 CA03BO 155551057 IC50 = 630.96 nM T68547 C4Q7CM 155551213 IC50 = 277 nM T68547 C3JQ1N 155551780 IC50 = 676 nM T68547 CE01AP 155551891 IC50 = 8.2 nM T68547 CEO4J8 155551917 IC50 = 10.31 nM T68547 C05ZVG 155552130 IC50 = 8.8 nM T68547 CV4Y5B 155552792 IC50 = 4200 nM T68547 CXT8F1 155552802 IC50 = 11000 nM T68547 CPML83 155553104 IC50 = 8360 nM T68547 CH6MF0 155553120 IC50 = 10.5 nM T68547 CMRJ52 155553215 IC50 = 2070 nM T68547 C7PBK3 155553376 IC50 = 280 nM T68547 CGDF76 155554360 IC50 = 8100 nM T68547 CXGE59 155554383 IC50 = 27 nM T68547 CC56ED 155554844 IC50 = 4.2 nM T68547 CXGR50 155555191 IC50 = 24800 nM T68547 C9DPQ1 155555248 IC50 = 7200 nM T68547 C8ZD2Y 155555330 IC50 = 1300 nM T68547 CT7GW1 155555345 IC50 = 100 nM T68547 CZ5OP3 155555490 IC50 = 2150 nM T68547 CFW90N 155555562 IC50 = 0.21 nM T68547 CE5P4I 155555900 IC50 = 47 nM T68547 C7QTU1 155555957 IC50 > 50000 nM T68547 CWV2Y0 155556131 IC50 = 39 nM T68547 CIN57Q 155556138 IC50 = 896 nM T68547 C6IL1E 155557199 IC50 = 28.84 nM T68547 C0IO1Q 155557341 IC50 = 32 nM T68547 CNM71L 155557418 IC50 = 216.5 nM T68547 CTL5E3 155557538 IC50 = 125 nM T68547 CN32AF 155557637 IC50 = 6420 nM T68547 CU78QC 155557817 IC50 > 1000 nM T68547 C8AUB0 155558567 IC50 = 65.1 nM T68547 CK3B2T 155558642 IC50 = 1900 nM T68547 CX70UY 155558767 IC50 = 1.3 nM T68547 C9Q6MF 155558959 IC50 = 28 nM T68547 C6N2VW 155559068 IC50 = 690 nM T68547 C2IS1E 155559200 IC50 = 8.71 nM T68547 CPD50Q 155559583 IC50 = 3500 nM T68547 CBYQ06 155559698 IC50 = 8210 nM T68547 CU2Y5S 155559868 IC50 = 3.5 nM T68547 CC62UI 155559872 IC50 = 57 nM T68547 CQ46GB 155559916 IC50 = 147.5 nM T68547 C57LYD 155560018 IC50 = 73 nM T68547 CMD6Q7 155560250 IC50 = 2380 nM T68547 CZX9P3 155560271 IC50 = 0.11 nM T68547 CGH85A 155560338 IC50 = 3.3 nM T68547 CT31YW 155560779 IC50 = 2300 nM T68547 CID3V4 155560946 IC50 = 5020 nM T68547 CW50YA 155561265 IC50 = 180.9 nM T68547 CQ0T4D 155561330 IC50 = 91 nM T68547 C1QZ8A 155561726 IC50 = 1.8 nM T68547 CJPL17 155561829 IC50 = 21.2 nM T68547 CJ4KO7 155562145 IC50 = 87.98 nM T68547 CGL24S 155562249 IC50 = 17700 nM T68547 CC6H1B 155562568 IC50 = 0.82 nM T68547 CSJ23C 155562809 IC50 = 449 nM T68547 CBJ03Y 155563284 IC50 = 463 nM T68547 CXEQ27 155563524 IC50 = 1000 nM T68547 CBJ58X 155563536 IC50 = 167 nM T68547 CXWU93 155563558 IC50 = 100 nM T68547 C9UYZ6 155564157 IC50 = 5.929 nM T68547 CX23YB 155564400 IC50 = 78.5 nM T68547 CFH0O8 155564436 IC50 = 3080 nM T68547 CR85ZW 155564587 IC50 = 1670 nM T68547 C8P5ZA 155564733 IC50 = 134.1 nM T68547 CPNA06 155564750 IC50 > 50000 nM T68547 C87JXN 155564870 IC50 = 794.33 nM T68547 CAG01V 155565290 IC50 = 847 nM T68547 C7P5NL 155565471 IC50 = 73 nM T68547 CZDC03 155565491 IC50 > 30000 nM T68547 CG65CR 155565674 IC50 = 50000 nM T68547 C2IVK7 155565738 IC50 = 27.8 nM T68547 CKJ36M 155565775 IC50 = 84 nM T68547 CD05RS 155566122 IC50 > 50000 nM T68547 C4A0RK 155566461 IC50 > 50000 nM T68547 C51BFK 155566644 IC50 = 51 nM T68547 CP1MH4 155566833 IC50 = 2400 nM T68547 C6V3EC 155567228 IC50 = 2.1 nM T68547 C6DQ2X 155567318 IC50 = 37 nM T68547 C04CGS 155567444 IC50 > 50000 nM T68547 CT6Z4H 155567814 IC50 = 2.189 nM T68547 C7RBT1 155567880 IC50 = 2.2 nM T68547 CA7B0F 155568022 IC50 = 2240 nM T68547 CS03PJ 155568350 IC50 > 50000 nM T68547 CX9V3D 155568494 IC50 > 30000 nM T68547 C19YAS 155568707 IC50 = 5720 nM T68547 CF2X0U 155568767 IC50 = 290 nM T68547 C46XEM 155568884 IC50 = 19 nM T68547 C3W7RP 155569171 IC50 = 281 nM T68547 C0RNZ1 155569208 IC50 = 872 nM T68547 C5NQK8 155569352 IC50 = 0.9177 nM T68547 CW5XB4 155569484 IC50 = 2490 nM T68547 CQ6C3M 155569679 IC50 = 30 nM T68547 C3BAZ5 24861442 IC50 = 9 nM T68547 CZVT07 44422818 IC50 = 40000 nM T68547 D00GBB 11449246 Ki = 16 nM T68547 D00HFS 46884057 IC50 = 76 nM T68547 D00HXX 56650312 IC50 = 5600 nM T68547 D00KFF 9882812 IC50 = 7800 nM T68547 D00LSZ 11044829 IC50 = 35 nM T68547 D00PLM 44418106 IC50 = 1130 nM T68547 D00RGD 11128726 IC50 = 153 nM T68547 D00SEE 11379392 IC50 = 218 nM T68547 D00XTC 44437872 IC50 = 36 nM T68547 D01BCK 23382 IC50 > 100000 nM T68547 D01DOV 23634888 IC50 = 52300 nM T68547 D01EDB 135903324 IC50 = 104 nM T68547 D01FYB 23648267 IC50 = 2000 nM T68547 D01YBR 44591988 IC50 = 3060 nM T68547 D02HVH 11427204 IC50 = 48 nM T68547 D02NAF 44437870 IC50 = 2.7 nM T68547 D02NVY 44437869 IC50 = 2 nM T68547 D02NWS 279980 Ki = 295 nM T68547 D02VVU 44328873 EC50 = 5000 nM T68547 D03FFI 11129854 IC50 = 35 nM T68547 D03FOD 21397854 IC50 = 715 nM T68547 D03HNC 17748273 IC50 > 100000 nM T68547 D03OYL 16655084 IC50 = 0.9 nM T68547 D03PRG 44437878 IC50 = 5.3 nM T68547 D03QOD 239512 IC50 > 10000 nM T68547 D03ZUZ 11381650 IC50 = 8280 nM T68547 D04CDZ 44437873 IC50 = 170 nM T68547 D04DOL 25032059 IC50 = 33 nM T68547 D04KQF 6675804 Ki = 28 nM T68547 D04UVL 1133083 IC50 = 2600 nM T68547 D04XPZ 11822609 IC50 = 8 nM T68547 D05OVV 11993691 IC50 = 730 nM T68547 D05PYF 10242569 IC50 = 243 nM T68547 D05QBX 44369352 IC50 > 100000 nM T68547 D06FAK 46918725 IC50 = 3074 nM T68547 D06NVX 25002768 IC50 = 900 nM T68547 D07HUH 44418155 IC50 = 18.8 nM T68547 D07YZZ 5173 Ki = 19 nM T68547 D08XMS 44591267 IC50 = 9 nM T68547 D09RKA 72946782 IC50 = 5000 nM T68547 D0A6CB 10314237 IC50 = 5 nM T68547 D0A7IF 44418125 IC50 = 1260 nM T68547 D0B1YM 135894458 IC50 = 10900 nM T68547 D0B3ZM 11436024 IC50 = 791 nM T68547 D0CJ7L 10891349 IC50 = 6 nM T68547 D0D3XC 11708207 IC50 = 670 nM T68547 D0E0TA 44454650 IC50 = 58 nM T68547 D0E8UH 44437879 IC50 = 3.2 nM T68547 D0E9DD 16095101 IC50 = 50 nM T68547 D0G0OF 44418145 IC50 = 3.6 nM T68547 D0G1EX 44437876 IC50 = 88 nM T68547 D0G3ZH 25216936 IC50 > 10000 nM T68547 D0GJ1E 11120992 IC50 = 45 nM T68547 D0H4YW 3611 Ki > 2500 nM T68547 D0H7QA 46884056 IC50 = 57 nM T68547 D0K7QR 45269423 IC50 = 140 nM T68547 D0K8MF 10858374 IC50 = 450 nM T68547 D0KM7H 11821974 IC50 = 95 nM T68547 D0L4ML 11031415 IC50 = 1500 nM T68547 D0L5WI 11833001 IC50 = 25 nM T68547 D0L6YF 46884016 IC50 = 71 nM T68547 D0M0QJ 10452725 IC50 = 29 nM T68547 D0M1ZI 16095112 IC50 = 1830 nM T68547 D0M9LJ 44454415 IC50 = 48 nM T68547 D0MC9C 50908800 IC50 = 1420 nM T68547 D0MD7H 44454143 IC50 = 52 nM T68547 D0N5RV 44437875 IC50 = 4.7 nM T68547 D0N9AK 44138031 IC50 = 5480 nM T68547 D0O7UF 10923922 IC50 = 15 nM T68547 D0P1RQ 9924962 IC50 = 1000 nM T68547 D0PP3Q 44418185 IC50 = 2500 nM T68547 D0Q2CC 46884055 IC50 = 576 nM T68547 D0Q2GM 44454416 IC50 = 65 nM T68547 D0Q4AV 25216938 IC50 > 10000 nM T68547 D0Q4EG 4882 IC50 > 180000 nM T68547 D0Q5DI 71462653 IC50 = 360 nM T68547 D0Q5MC 24753719 IC50 = 3800 nM T68547 D0Q8QA 44418141 IC50 = 750 nM T68547 D0Q9PO 16095114 Ki = 20 nM T68547 D0QX6R 10998964 IC50 = 500 nM T68547 D0R3XO 44437883 IC50 = 94 nM T68547 D0R8JK 25216937 IC50 > 10000 nM T68547 D0S0WK 11075845 IC50 = 65 nM T68547 D0T0BE 11426781 IC50 = 145 nM T68547 D0T0SK 44138032 IC50 = 790 nM T68547 D0T4JQ 264 IC50 = 16000 nM T68547 D0T8AJ 23634372 IC50 > 10000 nM T68547 D0U0EZ 44437880 IC50 = 6.4 nM T68547 D0U3MB 9888071 IC50 = 1 nM T68547 D0U8FC 759408 IC50 = 2400 nM T68547 D0V1HA 24880249 IC50 > 100000 nM T68547 D0W1PV 6918328 Ki = 0.04 nM T68547 D0X1CB 395803 IC50 = 0.11 nM T68547 D0X4QC 44437877 IC50 = 6.2 nM T68547 D0X4VO 44359538 IC50 = 30000 nM T68547 D0XU0G 44591342 IC50 > 10000 nM T68547 D0XZ9Q 11149404 IC50 = 294 nM T68547 D0YO6M 785232 IC50 = 2000 nM T68547 D0YP4F 10383069 IC50 = 3 nM T68547 D0Z2VP 11139963 IC50 = 135 nM T68547 D0Z6HR 44437874 IC50 = 3.7 nM T68547 D0Z6MI 44437868 IC50 = 3.9 nM T68547 D0Z8PX 24757913 IC50 = 10.09 nM T48069 D01PZD 5329098 IC50 > 10000 nM T48069 D03ZBT 11626560 IC50 = 143 nM T48069 D04LVK 57379345 IC50 = 410 nM T48069 D07POC 176870 IC50 > 30000 nM T48069 D08CDI 208908 IC50 > 30000 nM T48069 D08PIE 68165256 IC50 = 24.9 nM T48069 D0E6XR 3062316 IC50 > 50000 nM T48069 D0G6QF 3081361 IC50 > 10000 nM T48069 D0IQ6P 25102847 IC50 > 10000 nM T48069 D0K8KX 5280343 IC50 = 300 nM T48069 D0O8GK 71496458 IC50 = 2900000 nM T48069 D01GFX 11640390 IC50 = 13 nM T48069 D02NNV 3038525 IC50 > 5000 nM T48069 D02QWY 24785538 IC50 = 1.8 nM T48069 D02UFQ 11620908 IC50 > 10000 nM T48069 D03LWG 53235510 IC50 > 10000 nM T48069 D07EHV 44814409 IC50 > 10000 nM T48069 D07HPJ 11476171 IC50 = 60 nM T48069 D08HOM 46207586 IC50 = 539 nM T48069 D0E3TC 44259 IC50 = 35.03 nM T48069 D0O0LS 25141092 IC50 = 122 nM T48069 D0O9PQ 57390074 IC50 = 3.2 nM T48069 D0P1CV 46191454 IC50 > 10000 nM T48069 D0P6DJ 151194 IC50 > 10000 nM T48069 D0Q7RE 16007391 Ki > 10000 nM T48069 D0Q9UX 16718576 IC50 > 10000 nM T48069 D0S5RC 3025986 IC50 > 25000 nM T48069 D03BNU 59604787 IC50 > 10000 nM T48069 D0LF0O 135441202 IC50 = 34 nM T48069 D0DK4I 4534 IC50 = 900 nM T48069 D0YK9D 9956119 IC50 > 10000 nM T48069 D04FHB 6918852 Ki > 5000 nM T48069 D0L5YF 5329032 IC50 > 20000 nM T48069 D0T3ME 156422 IC50 > 30000 nM T48069 C97TNH 10177 IC50 > 1000000 nM T48069 C63WLY 89644 IC50 = 3.5 ug.mL-1 T48069 CE4K5D 92516 IC50 > 50000 nM T48069 C5JE2Z 104860 IC50 = 1.7 ug.mL-1 T48069 C6Y9CV 151193 IC50 > 10000 nM T48069 CI1NA5 159926 IC50 > 10 ug.mL-1 T48069 CI80NA 160436 IC50 > 50000 nM T48069 CYBA43 177458 IC50 = 2.8 ug.mL-1 T48069 C1UAQ4 342168 IC50 > 100000 nM T48069 C1ZG2U 449087 IC50 > 10000 nM T48069 C9D7UY 727518 IC50 > 100000 nM T48069 CXB5A2 964113 IC50 > 100000 nM T48069 C2VRY5 1204889 IC50 = 3300 nM T48069 CXBF05 1204893 IC50 = 400 nM T48069 CFN1X5 1205024 IC50 = 3300 nM T48069 C07AHW 1205040 IC50 = 5300 nM T48069 CKNO43 1205381 IC50 = 57 nM T48069 C9H7DW 1205672 IC50 = 61 nM T48069 C5PDS4 1206018 IC50 = 11100 nM T48069 CYG3F7 1206240 IC50 = 3400 nM T48069 C8TM4R 1206252 IC50 = 6700 nM T48069 C59JUN 1206254 IC50 = 2900 nM T48069 CAM8U9 1206256 IC50 = 1600 nM T48069 CSN92F 1206261 IC50 = 8800 nM T48069 CLAH32 1206264 IC50 = 11100 nM T48069 C0H3WZ 1206279 IC50 = 8600 nM T48069 CGK27H 1210312 IC50 > 100000 nM T48069 C43DZV 1214096 IC50 > 100000 nM T48069 CPV94W 1218955 IC50 = 250 nM T48069 C6IZE0 1225146 IC50 = 280 nM T48069 CY17ZI 1227452 IC50 = 1600 nM T48069 CRC01U 1227456 IC50 > 100000 nM T48069 C9ZW7G 1230091 IC50 = 15000 nM T48069 C90KON 1231530 IC50 = 10000 nM T48069 C3UT1Y 1232220 IC50 = 49800 nM T48069 C1I2UP 1232262 IC50 = 6300 nM T48069 C1VZ8Q 1232267 IC50 > 100000 nM T48069 CC5PW9 1232669 IC50 > 100000 nM T48069 C5TSE1 1232814 IC50 = 16800 nM T48069 C9Y0JC 1237187 IC50 = 6600 nM T48069 CDB17F 1538822 IC50 = 10000 nM T48069 CON65H 1565908 IC50 = 4900 nM T48069 CBV04C 1731052 IC50 = 8200 nM T48069 CG1FL5 1731078 IC50 = 5200 nM T48069 CPVD46 1774817 IC50 = 6300 nM T48069 CJ31FK 1810679 IC50 > 100000 nM T48069 C3DV8H 1810702 IC50 > 100000 nM T48069 C06VDC 1922265 IC50 > 100000 nM T48069 CY0EX9 2226536 IC50 > 100000 nM T48069 CZ2B4M 2358462 IC50 > 100000 nM T48069 CXA1L7 2365265 IC50 > 100000 nM T48069 CEF62M 2379240 IC50 > 100000 nM T48069 CKT64G 2396126 IC50 > 10000 nM T48069 C8F6DW 2716301 IC50 > 100000 nM T48069 CNZO64 2716309 IC50 > 100000 nM T48069 CM1A0Q 2766999 IC50 = 1308 nM T48069 C83SZF 2767000 IC50 = 2471 nM T48069 C6EY0A 2767002 IC50 = 1641 nM T48069 C3C7WT 2767003 IC50 = 34 nM T48069 C1FPC5 3074368 IC50 = 568 nM T48069 CCN9D5 3142817 IC50 = 310 nM T48069 CEL1J5 3524522 IC50 > 30000 nM T48069 C0LY1H 4269048 IC50 > 100000 nM T48069 C8IAR2 5281657 IC50 = 33300 nM T48069 CI68PW 5283685 IC50 = 2460 nM T48069 CXK0S6 5283727 IC50 = 2770 nM T48069 C15WJX 5288527 IC50 = 1260 nM T48069 CY28LS 5293755 IC50 > 100000 nM T48069 CZIU69 5304328 IC50 > 100000 nM T48069 CDQ3M7 5359485 IC50 = 1 ug.mL-1 T48069 C54BYP 5360741 IC50 = 1.7 ug.mL-1 T48069 CD65JT 5427216 IC50 > 100000 nM T48069 CPB95V 5427224 IC50 > 100000 nM T48069 CA6L5V 5707304 IC50 > 100000 nM T48069 C43YGE 5713379 IC50 > 100000 nM T48069 C7GD1T 5753500 IC50 = 1710 nM T48069 CT8U7I 5874584 IC50 > 100000 nM T48069 CM8LW9 6036100 IC50 > 100000 nM T48069 CEOT94 6155669 IC50 = 6400 nM T48069 CQ3S8L 6450842 IC50 > 100000 nM T48069 CW5YJ2 6536705 IC50 > 100000 nM T48069 CQR03O 7117329 IC50 = 63000 nM T48069 C4G9WR 9547398 IC50 > 100000 nM T48069 C76CUP 9547698 IC50 = 2420 nM T48069 C2OL7K 9796455 IC50 >> 10000 nM T48069 C1E2DV 9826083 IC50 > 10000 nM T48069 C12PKF 9871380 IC50 > 25000 nM T48069 CUZ07T 9884745 IC50 = 49500 nM T48069 CXA5C8 9893493 IC50 > 25000 nM T48069 C3VG9B 9902671 IC50 = 40 nM T48069 CPQ13K 9933545 IC50 = 20000000 nM T48069 C6HP3L 9948410 IC50 > 100000 nM T48069 CJL7H1 9965947 IC50 = 490 nM T48069 COQ24E 9967928 IC50 = 55 nM T48069 CO4N3Q 9995374 IC50 > 100000 nM T48069 C26QHZ 10005638 IC50 > 10000 nM T48069 CR8DA1 10024683 IC50 > 100000 nM T48069 CLA93G 10047202 IC50 = 2300 nM T48069 C3LCH5 10047545 IC50 > 100000 nM T48069 C7YD1X 10048045 IC50 > 25000 nM T48069 CCK25W 10070969 IC50 = 39100 nM T48069 C1JUF8 10073832 IC50 > 25000 nM T48069 CR3N8E 10109869 IC50 = 6458 nM T48069 CPY3Z4 10135786 IC50 = 3.3 nM T48069 C59FGN 10165455 IC50 > 1000 nM T48069 CC78NE 10179293 IC50 = 2.5 nM T48069 CN1V3T 10202829 IC50 = 2.4 nM T48069 CGOT91 10207821 IC50 > 100000 nM T48069 C5YCN2 10215023 IC50 > 100000 nM T48069 CSHK19 10222816 IC50 = 5.2 nM T48069 CPD6Z9 10236164 IC50 > 100000 nM T48069 CSGD16 10246246 IC50 > 7000 nM T48069 CMX73A 10257575 IC50 = 300 nM T48069 CBI47E 10264222 IC50 > 100000 nM T48069 C0UOJ3 10270679 IC50 = 507 nM T48069 CJGH26 10275985 IC50 = 81 nM T48069 C7SFI1 10296883 IC50 > 10000 nM T48069 CR26KQ 10297734 IC50 = 847 nM T48069 C1AKH9 10303277 IC50 = 66 nM T48069 CA8B5T 10390073 IC50 > 10000 nM T48069 CBST19 10392387 IC50 = 150 nM T48069 CU49NB 10414315 IC50 = 600 nM T48069 C4CP7K 10423452 IC50 = 8600 nM T48069 CQ43JU 10426229 IC50 = 10100 nM T48069 C7HBP6 10429593 IC50 > 10000 nM T48069 CQIX92 10459386 IC50 = 151 nM T48069 C7PLI5 10478569 IC50 > 25000 nM T48069 CJWH60 10489322 IC50 > 100000 nM T48069 C5SVT4 10537949 IC50 > 100000 nM T48069 CGAW17 10562306 IC50 > 100000 nM T48069 C6AJI9 10562777 IC50 > 100000 nM T48069 CE5L6D 10587839 IC50 > 100000 nM T48069 CM8N6L 10593765 IC50 = 67600 nM T48069 CI30LZ 10613858 IC50 > 100000 nM T48069 CH6Z3L 10635478 IC50 > 100000 nM T48069 CB97UD 10636005 IC50 > 100000 nM T48069 C2UWA0 10658651 IC50 > 100000 nM T48069 C5L0IX 10663368 IC50 > 100000 nM T48069 C9Z7XH 10663503 IC50 > 100000 nM T48069 CH1G6P 10682457 IC50 > 100000 nM T48069 CP9XE8 10686611 IC50 > 100000 nM T48069 C83QWV 10714343 IC50 = 11800 nM T48069 C54UAK 10728035 IC50 > 100000 nM T48069 CXSH91 10753550 IC50 > 100000 nM T48069 CVPW04 10755069 IC50 > 100000 nM T48069 C3WR0Q 10779668 IC50 > 100000 nM T48069 CF5T1H 10783444 IC50 > 100000 nM T48069 C0KD7L 10805173 IC50 > 100000 nM T48069 C29IEM 11153568 IC50 = 1680 nM T48069 C8G5WP 11210533 IC50 = 150 nM T48069 CGO2Y1 11225122 IC50 = 398 nM T48069 C2W5RC 11235063 IC50 > 50000 nM T48069 CM4NY6 11236085 IC50 > 10000 nM T48069 C5OP0M 11269934 IC50 = 526 nM T48069 CUO27S 11282791 IC50 > 2000 nM T48069 CVA1O4 11292513 IC50 = 1350 nM T48069 CBOP58 11293798 Ki > 10000 nM T48069 CX49HY 11306193 IC50 = 547 nM T48069 CSU4H3 11338098 IC50 = 1050 nM T48069 C2R6DG 11350054 IC50 = 3510 nM T48069 CK49IR 11361235 IC50 = 1230 nM T48069 C57VFQ 11361434 IC50 > 10000 nM T48069 C26BZX 11362471 Ki > 10000 nM T48069 CB4JW0 11385175 IC50 = 775 nM T48069 CWXB93 11397177 Ki > 10000 nM T48069 CM5S7I 11408442 IC50 = 105 nM T48069 C7AI2V 11432911 IC50 > 25000 nM T48069 C7ZR9K 11442386 IC50 = 116 nM T48069 C9M2GF 11464085 IC50 = 3790 nM T48069 C35MVJ 11471056 IC50 > 10000 nM T48069 CU2Q0H 11476255 IC50 > 10000 nM T48069 C6M9NC 11477626 IC50 > 25000 nM T48069 C0DP8R 11494064 IC50 = 1040 nM T48069 C80CMJ 11502053 IC50 = 270 nM T48069 CR2Z8J 11504226 IC50 = 651 nM T48069 CL7X4Q 11530963 IC50 = 6967 nM T48069 CACS26 11561968 Ki > 2000 nM T48069 CO9KP5 11583459 IC50 = 20 nM T48069 CF58CN 11604324 IC50 = 166 nM T48069 C43JZU 11604436 IC50 = 15000 nM T48069 CGU7N0 11604739 IC50 > 20000 nM T48069 C5B3XJ 11620410 IC50 = 4010 nM T48069 CSM62L 11626920 IC50 > 30000 nM T48069 CN4R5G 11632540 IC50 = 86 nM T48069 CK34LS 11632737 IC50 > 25000 nM T48069 CU38TK 11649146 IC50 = 14 nM T48069 CAJS96 11662893 IC50 > 20000 nM T48069 CKAH36 11669784 IC50 = 7000 nM T48069 CS4R8Z 11670378 IC50 = 17 nM T48069 CU0E8O 11690457 Ki > 2000 nM T48069 C1OI3P 11690914 IC50 = 19 nM T48069 C5RWO2 11716093 IC50 = 518 nM T48069 C7WMH2 11716669 IC50 > 10000 nM T48069 C45EWD 11723489 IC50 > 7000 nM T48069 CG2NR5 11750704 IC50 = 119 nM T48069 C62YLE 11758149 IC50 = 460 nM T48069 C1ITY8 11773105 IC50 = 606 nM T48069 CS36BH 11843159 IC50 > 25000 nM T48069 C8NF6H 11947782 Ki = 887 nM T48069 CO8QR4 11962890 Ki = 1570 nM T48069 C0HE1D 11962891 Ki = 26.5 nM T48069 CFP7M5 11962976 Ki = 1290 nM T48069 CP89KY 11962977 Ki = 104 nM T48069 CCY4J2 11962978 Ki = 70.2 nM T48069 C3XWU1 11963015 Ki = 872 nM T48069 CA7Y5P 11963057 Ki = 1100 nM T48069 CTC31Z 11963059 Ki = 419 nM T48069 C3H4PA 11963103 Ki = 249 nM T48069 CI7G5W 11963258 Ki = 928 nM T48069 CT1RA7 11963259 Ki > 6600 nM T48069 CY8GD6 11963300 Ki = 1800 nM T48069 CQ2WD1 11963302 Ki = 744 nM T48069 CGCX39 11963344 Ki = 35.9 nM T48069 C4O3UR 11963386 Ki = 18.5 nM T48069 CPG89E 11963387 Ki = 144 nM T48069 CF3W2N 11963388 Ki = 42.7 nM T48069 CQT2I1 11963389 Ki = 24.8 nM T48069 CT91NG 11963423 Ki = 30.9 nM T48069 CH2A1C 11963425 Ki = 87.7 nM T48069 C87DIW 12758175 IC50 = 52000 nM T48069 C7Y1XF 14852609 IC50 = 600 nM T48069 C1YO9X 15135539 IC50 = 800 nM T48069 CDGF78 15282555 IC50 = 2300 nM T48069 C7LB4I 15949613 IC50 > 10000 nM T48069 CQR5O7 16042971 IC50 > 10000 nM T48069 C9TU1O 16046126 IC50 > 1000 nM T48069 CH9YP5 16085873 IC50 > 30000 nM T48069 CPT8G9 16085888 IC50 = 13900 nM T48069 COX7D2 16085894 IC50 > 30000 nM T48069 CQG45C 16109001 IC50 = 927 nM T48069 CTG36E 16126863 IC50 = 80 nM T48069 C5VPH9 16129448 IC50 = 1280 nM T48069 CL5IF2 16214946 IC50 = 19 nM T48069 CJ5KU9 16659012 IC50 = 170 nM T48069 C2IF3P 16678352 IC50 = 2720 nM T48069 C3IO1C 16679060 IC50 > 30000 nM T48069 CM0Z2P 16730088 IC50 = 3050 nM T48069 C0H8UN 16730109 IC50 > 25000 nM T48069 CR1E4C 16747763 IC50 = 14000 nM T48069 CU5Q9B 16757524 Ki = 887 nM T48069 CL9BQ6 17748275 IC50 = 25000 nM T48069 C5EH9K 20817080 IC50 = 160 nM T48069 C0ZUW6 20817086 IC50 = 812.83 nM T48069 CS6CL5 20817096 IC50 = 584 nM T48069 C3AI0N 20817111 IC50 = 12.5 nM T48069 CISW64 20826919 IC50 = 251 nM T48069 CGH76Y 20826920 IC50 = 123 nM T48069 C48ROB 20826930 IC50 = 36 nM T48069 C0R8SV 20826932 IC50 = 3377 nM T48069 CE46AO 20826938 IC50 = 201 nM T48069 C62MBU 20826947 IC50 = 198 nM T48069 C5RK0O 20826972 IC50 = 22 nM T48069 CL48NF 20826990 IC50 = 725 nM T48069 CNF7Q4 20826992 IC50 = 58 nM T48069 CH4B5K 21081523 IC50 > 5000 nM T48069 C25UKC 21081761 IC50 > 5000 nM T48069 CL81VC 21100709 IC50 = 100000 nM T48069 CZJT36 21704852 IC50 = 1000 nM T48069 C7DYL5 21995160 IC50 = 30 nM T48069 C7W9UI 22477349 IC50 = 33 nM T48069 C9QLP0 23133323 IC50 > 20000 nM T48069 C6JV7W 23400934 IC50 > 7000 nM T48069 CD5S7O 23401001 IC50 > 7000 nM T48069 C7F3UK 23536360 IC50 = 13 nM T48069 C9K2AI 23536542 IC50 = 41 nM T48069 CJ1O8K 23656213 IC50 = 1000 nM T48069 C5QX0K 23729342 IC50 = 125 nM T48069 CUO58X 23729343 IC50 = 2322 nM T48069 CR0V7I 23729345 IC50 = 2794 nM T48069 CL2Z1P 23729346 IC50 = 35 nM T48069 C2RV3U 24180608 IC50 > 30000 nM T48069 CA3I4T 24753787 IC50 > 50000 nM T48069 C7YG1N 24759534 IC50 > 100000 nM T48069 CAJ4T2 24762205 IC50 > 10000 nM T48069 CQNP54 24764449 IC50 = 1000 nM T48069 CCPS81 24764502 IC50 > 35000 nM T48069 C81GVC 24774737 IC50 = 5011.87 nM T48069 CN6B1L 24774912 IC50 = 10000 nM T48069 CGY19Z 24785273 IC50 = 3 nM T48069 C9D5UV 24785537 IC50 = 4 nM T48069 CA7XJ1 24785806 IC50 = 1 nM T48069 CIQ2F7 24785807 IC50 = 9 nM T48069 C3SU9E 24785809 IC50 = 2 nM T48069 CCP2M3 24822704 IC50 > 50000 nM T48069 C07MSJ 24825716 IC50 = 9 nM T48069 CFK2B9 24882503 IC50 > 10000 nM T48069 C43HWQ 24883287 IC50 > 10000 nM T48069 C8DA5Q 24883334 IC50 > 10000 nM T48069 C4V9GH 24894117 IC50 = 22000 nM T48069 CZ6KD4 24894886 IC50 = 8700 nM T48069 CB5TP8 24894992 IC50 = 7700 nM T48069 C32SUJ 24894993 IC50 = 18000 nM T48069 CN13JF 24899915 IC50 = 4.9 ug.mL-1 T48069 CBWR97 24899916 IC50 = 0.91 ug.mL-1 T48069 C9F2JD 24899917 IC50 > 10 ug.mL-1 T48069 C64MTI 24900160 IC50 = 2.4 ug.mL-1 T48069 CO2I6Q 24900161 IC50 = 3.6 ug.mL-1 T48069 CD08VO 24901691 Ki = 178 nM T48069 C0NCI3 24901692 Ki = 915 nM T48069 C59ICM 24901693 Ki = 744 nM T48069 C9WD7I 24901694 Ki = 695 nM T48069 CLZ23U 24951610 IC50 = 30000 nM T48069 CD5HQ0 24969301 IC50 > 10000 nM T48069 C4EG8R 24993189 IC50 > 10000 nM T48069 CBK82P 25011729 IC50 > 30000 nM T48069 C6N7KR 25032700 IC50 > 1000 nM T48069 CD7V3A 25101485 IC50 = 162 nM T48069 CJ32TF 25101637 IC50 = 11 nM T48069 CHQ96L 25101638 IC50 = 8400 nM T48069 C4OA5D 25113170 IC50 = 2 nM T48069 CT5NA4 25113180 IC50 = 140 nM T48069 CTV54O 25123227 IC50 > 10000 nM T48069 CG9LW7 25123829 IC50 = 2 nM T48069 CG3XC9 25124150 IC50 = 5 nM T48069 CO2IR5 25124816 Ki = 1.6 nM T48069 C6BWZ8 25145145 IC50 > 100 nM T48069 C78YWA 25145716 IC50 > 500 nM T48069 C8IX5P 25174241 IC50 = 271 nM T48069 CE6PB7 25175712 IC50 = 1441 nM T48069 CB1Z8N 25175860 IC50 = 1335 nM T48069 CIHB16 25175861 IC50 = 206 nM T48069 C04HDK 25176007 IC50 = 209 nM T48069 CT2K5R 25176014 IC50 = 28 nM T48069 C6G7RT 25176165 IC50 = 124 nM T48069 C81NBM 25176332 IC50 = 2112 nM T48069 CX0O5A 25178331 IC50 = 2300 nM T48069 CIG4H0 25178539 IC50 = 4000 nM T48069 CTED51 25186142 IC50 = 12589.25 nM T48069 CNG96H 25210579 IC50 > 10000 nM T48069 CM0T8S 25210970 IC50 = 10 nM T48069 CW30KM 25210971 IC50 < 0.2 nM T48069 CB3Z8Q 25210972 IC50 = 0.2 nM T48069 CEU0R6 25211574 IC50 = 0.5 nM T48069 C3SYO4 25211575 IC50 = 487 nM T48069 CG40OH 25211676 IC50 = 1 nM T48069 CXE16F 25218564 IC50 = 160 nM T48069 C3RH2Q 25218565 IC50 = 20 nM T48069 C20THL 25218566 IC50 = 8 nM T48069 C25DJY 25218567 IC50 = 13 nM T48069 CHM29R 25218568 IC50 = 13 nM T48069 CI78TL 25218569 IC50 = 13 nM T48069 CG29EY 25218570 IC50 = 6 nM T48069 C16ISR 25218571 IC50 = 25 nM T48069 C9FAL8 25218572 IC50 = 377 nM T48069 C9G2ZM 25218573 IC50 = 63 nM T48069 CB03GW 25218574 IC50 = 6 nM T48069 CC39RK 25218575 IC50 = 4 nM T48069 C0ZJ3O 25218576 IC50 = 2 nM T48069 CRM7N5 25218577 IC50 = 3 nM T48069 CR3KE8 25218578 IC50 = 50 nM T48069 C6T9AO 25218579 IC50 = 85 nM T48069 CGK1O0 25218580 IC50 = 1 nM T48069 C0S4UP 25218581 IC50 = 128 nM T48069 C89DVN 25218582 IC50 = 32 nM T48069 CLM18I 25218583 IC50 = 72 nM T48069 CBSY10 25218584 IC50 = 32 nM T48069 CDYZ78 25218585 IC50 = 8 nM T48069 CCL2O3 25218586 IC50 = 298 nM T48069 CR3UY7 25218587 IC50 = 4 nM T48069 CN5X1G 25218588 IC50 = 40 nM T48069 C04PGY 25218589 IC50 = 25 nM T48069 CD7KC4 25218590 IC50 = 16 nM T48069 C1ODR5 25218591 IC50 = 1 nM T48069 CYB58C 25218592 IC50 = 10 nM T48069 CO0RF6 25218593 IC50 = 5 nM T48069 CFL60D 25218594 IC50 = 1.6 nM T48069 CZW87R 25218595 IC50 = 1.6 nM T48069 CCOA65 25218596 IC50 = 20 nM T48069 C1KR3Q 25218597 IC50 = 0.6 nM T48069 CF4JQ2 25218598 IC50 = 0.8 nM T48069 CH3L5J 25218599 IC50 = 3.2 nM T48069 CYG30F 25218600 IC50 = 60 nM T48069 CP81DI 25218601 IC50 = 0.3 nM T48069 CFK35N 25218602 IC50 = 1.6 nM T48069 CVQ2S8 25218603 IC50 = 0.8 nM T48069 CSI96B 25218604 IC50 = 68 nM T48069 C0X6KT 25218605 IC50 = 50 nM T48069 C6DHV0 25218606 IC50 = 10000 nM T48069 CEH1L3 25218607 IC50 = 3.2 nM T48069 C63XFG 25218608 IC50 = 2 nM T48069 C5USY6 25218609 IC50 = 2 nM T48069 CUD29Z 25218610 IC50 = 1.6 nM T48069 CHAW52 25218611 IC50 = 4 nM T48069 CX9IV4 25218612 IC50 = 3700 nM T48069 CAF65T 25218613 IC50 = 71 nM T48069 CI3X8Z 25218614 IC50 = 0.9 nM T48069 C50FJO 25218615 IC50 = 1.3 nM T48069 CK53NQ 25218616 IC50 = 0.8 nM T48069 C87ISA 25218617 IC50 = 0.5 nM T48069 C0HEP7 25218618 IC50 = 5 nM T48069 CM5RS9 25218619 IC50 = 135 nM T48069 CA5J0T 25218620 IC50 = 6.3 nM T48069 CJ3QC0 25218621 IC50 = 16 nM T48069 CH4T1J 25218622 IC50 = 5 nM T48069 CY32AD 25218623 IC50 = 25 nM T48069 C8LXB1 25218685 IC50 = 64 nM T48069 C3PT8E 25218686 IC50 = 23 nM T48069 CY35SP 25218687 IC50 = 81 nM T48069 CR0FO4 25218688 EC50 = 711 nM T48069 CWNY70 25218689 EC50 = 143 nM T48069 CZ5M3A 25218690 EC50 = 247 nM T48069 CK9AO6 25218691 EC50 = 208 nM T48069 CXH7F8 25218692 EC50 = 115 nM T48069 CH2GL3 25218693 IC50 = 40 nM T48069 CSE42H 25218793 IC50 = 26 nM T48069 CR10HZ 25218794 IC50 = 65 nM T48069 CA8N3M 25218796 IC50 = 10 nM T48069 CL3K7N 25218797 IC50 = 30 nM T48069 CD1OX9 25218798 IC50 = 394 nM T48069 C1Q9CJ 25218799 IC50 = 13700 nM T48069 C5M4KZ 25218801 IC50 = 26 nM T48069 C8QW5N 25218802 IC50 = 3880 nM T48069 C7HNF6 25218803 IC50 = 24 nM T48069 C5ZLW1 25218804 IC50 = 30 nM T48069 CU82XS 25218805 IC50 = 45 nM T48069 CDT35X 25218806 IC50 = 32 nM T48069 C3XBV0 25218808 IC50 = 31 nM T48069 CZ0BK3 25218809 IC50 = 11 nM T48069 CAB96P 25218810 IC50 = 14 nM T48069 CH5W9G 25218811 IC50 = 20 nM T48069 CKU9B4 25218812 IC50 = 67 nM T48069 CQ1G3V 25218814 IC50 = 14 nM T48069 C8PA9Y 25218815 IC50 = 15 nM T48069 CAO7Z3 25218816 IC50 = 13 nM T48069 CP6VZ4 25218817 IC50 = 47 nM T48069 CY93GM 25218818 IC50 = 16 nM T48069 CLS98P 25218819 IC50 = 16 nM T48069 C19ZOE 25218820 IC50 = 189 nM T48069 CG43WC 25218821 IC50 = 79 nM T48069 CM2GY7 25218822 IC50 = 50 nM T48069 CD80NJ 25218823 IC50 = 88 nM T48069 CT84WC 25218824 IC50 > 10000 nM T48069 C1KI9V 25920884 IC50 = 14 nM T48069 CHO43Y 28491869 IC50 = 1690 nM T48069 CO8I0Q 42601408 IC50 = 0.5 nM T48069 C8T5IH 42602949 IC50 = 79432.82 nM T48069 CJ5U1X 42639664 IC50 = 1.9 ug.mL-1 T48069 C5PWI0 44129657 IC50 > 10000 nM T48069 CTN41Y 44156909 IC50 > 10000 nM T48069 CN0X1C 44156917 IC50 > 10000 nM T48069 CG41XM 44219728 IC50 = 21 nM T48069 CEL61X 44229839 IC50 > 10000 nM T48069 CSY8A3 44321301 IC50 > 100000 nM T48069 CCG2M5 44321317 IC50 > 100000 nM T48069 CY9ED1 44321395 IC50 > 100000 nM T48069 C5U1CR 44321686 IC50 > 10000 nM T48069 CETY53 44321717 IC50 > 100000 nM T48069 CV60ME 44321734 IC50 > 50000 nM T48069 C0KD4U 44346053 IC50 > 10000 nM T48069 CYV2D7 44368815 IC50 = 64000 nM T48069 CJT6H8 44438832 IC50 > 10000 nM T48069 CD7RZ6 44438834 IC50 > 10000 nM T48069 C1YEG7 44438836 IC50 = 1970 nM T48069 CO7PI2 44438839 IC50 > 10000 nM T48069 C53CMH 44438841 IC50 = 3500 nM T48069 CX6T4W 44438843 IC50 = 1050 nM T48069 C32CKD 44438844 IC50 = 2270 nM T48069 C0TMV8 44438845 IC50 = 1110 nM T48069 C5A0RK 44438850 IC50 = 6280 nM T48069 CRC6K9 44438853 IC50 > 10000 nM T48069 CF2LO4 44438854 IC50 > 10000 nM T48069 C7R2BJ 44438855 IC50 > 10000 nM T48069 C9RO2V 44438856 IC50 = 1090 nM T48069 CJL6B4 44438858 IC50 > 10000 nM T48069 CZC53O 44438860 IC50 = 2060 nM T48069 CP01ZL 44438862 IC50 = 510 nM T48069 CRD9T0 44438864 IC50 = 343 nM T48069 CD2OU7 44438866 IC50 = 2120 nM T48069 CRL0B9 44438867 IC50 = 980 nM T48069 C8Z1RL 44438873 IC50 = 3280 nM T48069 C48OVM 44438876 IC50 = 5780 nM T48069 CBN1H0 44438878 IC50 = 2820 nM T48069 CW15DA 44438882 IC50 > 10000 nM T48069 CD9W5S 44438883 IC50 = 898 nM T48069 CA52ML 44438887 IC50 = 4480 nM T48069 C9WP2R 44438890 IC50 = 329 nM T48069 CI0V8D 44438892 IC50 = 1590 nM T48069 C5XUK3 44438894 IC50 = 1350 nM T48069 CT51XC 44438896 IC50 = 1670 nM T48069 C8G2JP 44438898 IC50 = 248 nM T48069 CA6P4J 44438904 IC50 > 10000 nM T48069 CH4LQ6 44438909 IC50 > 10000 nM T48069 C0QPU2 44438923 IC50 = 1820 nM T48069 C15QMJ 44438924 IC50 = 3400 nM T48069 C8K9AZ 44438925 IC50 = 1300 nM T48069 CP36YS 44438928 IC50 = 1390 nM T48069 CRCP07 44438929 IC50 = 115 nM T48069 C8Y4OZ 44438931 IC50 = 60 nM T48069 C97ORA 44438933 IC50 = 346 nM T48069 CV8Q6L 44438937 IC50 = 148 nM T48069 C5J3IW 44438938 IC50 = 220 nM T48069 COB1X6 44438940 IC50 = 265 nM T48069 C3M0KB 44440174 IC50 = 800 nM T48069 C74DFE 44440176 IC50 = 1000 nM T48069 CU8L9H 44440177 IC50 = 800 nM T48069 C3SRV6 44440179 IC50 = 1000 nM T48069 C4J6AM 44440180 IC50 = 1100 nM T48069 C48PXY 44441698 IC50 = 787 nM T48069 CE15CH 44441699 IC50 = 487 nM T48069 C2CE8L 44441700 IC50 = 38 nM T48069 C1LIN5 44441702 IC50 = 168 nM T48069 CVG1N0 44441706 IC50 = 65 nM T48069 CCO78B 44441707 IC50 = 123 nM T48069 C26USE 44441709 IC50 = 186 nM T48069 CNS92V 44441711 IC50 = 140 nM T48069 C3AI2P 44441712 IC50 = 642 nM T48069 C92PUE 44441714 IC50 = 70 nM T48069 CXS1Y4 44441715 IC50 = 1250 nM T48069 C50UFA 44441717 IC50 = 104 nM T48069 CJIP27 44441719 IC50 = 90 nM T48069 CJV84M 44441720 IC50 = 152 nM T48069 C2WDZ7 44441722 IC50 = 173 nM T48069 C0TC7N 44441723 IC50 = 674 nM T48069 CYF6Z8 44441726 IC50 = 429 nM T48069 C6BU0O 44441728 IC50 = 32 nM T48069 C1QW3X 44441730 IC50 = 2337 nM T48069 CCS1N3 44441733 IC50 = 1309 nM T48069 C6R4NV 44441735 IC50 = 1542 nM T48069 C4Y8XV 44446930 IC50 > 1000 nM T48069 CWBV18 44446940 IC50 = 360 nM T48069 CPR51F 44446941 IC50 = 700 nM T48069 CQ28KT 44451337 IC50 > 10000 nM T48069 CTLO32 44451459 IC50 = 18 nM T48069 CW62HN 44451470 IC50 = 47 nM T48069 C7WM5I 44451471 IC50 = 130 nM T48069 CXRG25 44451484 IC50 = 77 nM T48069 C4U8SK 44451494 IC50 = 147 nM T48069 CZB82I 44451497 IC50 = 148 nM T48069 C7HIM2 44452543 IC50 > 2000 nM T48069 CZ9H4D 44452544 IC50 > 2000 nM T48069 CN40UR 44480282 IC50 = 291 nM T48069 C4B7KF 44515722 IC50 = 12.8 nM T48069 C8H4FA 44515723 IC50 = 139 nM T48069 CYH6P3 44520205 IC50 > 10000 nM T48069 C3Q0DX 44564789 IC50 = 1500 nM T48069 CP40XB 44564790 IC50 = 3600 nM T48069 C35NTB 44564791 IC50 = 4400 nM T48069 CJY83G 44564817 IC50 = 2900 nM T48069 CLK98G 44564818 IC50 > 10000 nM T48069 CF2D1K 44564819 IC50 > 10000 nM T48069 C3CQ9K 44564820 IC50 > 10000 nM T48069 CI8V2L 44564821 IC50 > 10000 nM T48069 C9PO7J 44564860 IC50 > 10000 nM T48069 C16FJW 44564861 IC50 > 10000 nM T48069 C8AMX5 44564862 IC50 = 860 nM T48069 CTR59U 44564863 IC50 > 10000 nM T48069 C9EY4C 44564864 IC50 = 800 nM T48069 CG5Z7T 44564910 IC50 = 1100 nM T48069 CU9O4C 44564911 IC50 = 3300 nM T48069 CXZ15S 44564954 IC50 > 10000 nM T48069 CZ78WJ 44564955 IC50 = 1650 nM T48069 CJ1X9V 44565013 IC50 = 100 nM T48069 CN2Q3D 44565014 IC50 = 810 nM T48069 CM2GN3 44565015 IC50 > 10000 nM T48069 C6RV9I 44565016 IC50 = 1200 nM T48069 CJC85A 44565069 IC50 = 7500 nM T48069 C8TLA3 44569603 IC50 = 1090 nM T48069 CQ72ZN 44569674 IC50 = 20 nM T48069 CIDV31 44569742 IC50 = 135 nM T48069 CK15QH 44569743 IC50 = 17 nM T48069 C0I1HE 44571763 IC50 = 2 nM T48069 CJT87P 44571764 IC50 = 5930 nM T48069 CZU40I 44571765 IC50 = 10 nM T48069 CSA56C 44571766 IC50 = 440 nM T48069 CF29RC 44571808 IC50 = 509 nM T48069 C6N8VZ 44571809 IC50 = 7 nM T48069 CISJ12 44571810 IC50 = 1 nM T48069 C90EIF 44571811 IC50 = 4 nM T48069 CQZ25P 44571812 IC50 = 1 nM T48069 CKE8N1 44571813 IC50 = 2 nM T48069 CXZ8C5 44571814 IC50 = 2 nM T48069 CR28WX 44571815 IC50 = 2 nM T48069 CX6Y8H 44571816 IC50 = 2 nM T48069 C5LDI7 44571817 IC50 = 2 nM T48069 CB0FH9 44571818 IC50 = 4 nM T48069 CIN37B 44571819 IC50 = 3 nM T48069 CWFB42 44571820 IC50 = 7 nM T48069 COLB09 44581217 IC50 = 654 nM T48069 C0DM5B 44581218 IC50 = 1.6 nM T48069 CX9B8I 44581220 IC50 = 1.3 nM T48069 CL9B8I 44581221 IC50 = 9 nM T48069 C9L8IT 44581222 IC50 = 0.8 nM T48069 C6DYT9 44581223 IC50 = 0.7 nM T48069 CCU1E3 44581247 IC50 = 0.5 nM T48069 CT0R7C 44581248 IC50 = 0.8 nM T48069 CD1R5B 44581270 IC50 = 2 nM T48069 C27HSX 44581271 IC50 = 28 nM T48069 C0EDL8 44581728 IC50 = 79 nM T48069 CN7OF6 44581729 IC50 = 32 nM T48069 C17CMQ 44581764 IC50 = 13 nM T48069 CRG26Q 44581766 IC50 = 400 nM T48069 CN4GM7 44597056 IC50 = 41 nM T48069 CRZ19V 44597164 IC50 = 199 nM T48069 C0HLQ5 44597165 IC50 = 13 nM T48069 C6ZX3F 44597166 IC50 = 40 nM T48069 CRE4X5 44597167 IC50 = 717 nM T48069 C98RLO 44597168 IC50 = 6 nM T48069 CU3RF1 45139989 IC50 > 10000 nM T48069 CQGZ06 45139991 IC50 > 10000 nM T48069 CM6BL0 45266936 IC50 = 242 nM T48069 C4K8BX 45267171 IC50 = 24700 nM T48069 C25VIM 45267176 IC50 = 11800 nM T48069 C0QH1J 45267792 IC50 = 335 nM T48069 CQV67O 45267795 IC50 = 1041 nM T48069 C8W5MA 45267796 IC50 = 3623 nM T48069 CIX1D3 45268678 IC50 = 57 nM T48069 CAJ1E5 45268679 IC50 = 31 nM T48069 CC61YO 45268681 IC50 = 64 nM T48069 C3LP8I 45269539 IC50 = 605 nM T48069 C3P1VD 45269546 IC50 = 3071 nM T48069 C9FJD6 45270367 IC50 = 200 nM T48069 C2JVA4 45270368 IC50 = 50 nM T48069 CQGS80 45270369 IC50 = 67 nM T48069 C8J5RI 45270370 IC50 = 127 nM T48069 CF60UQ 45270372 IC50 = 233 nM T48069 C59MTR 45270373 IC50 = 407 nM T48069 CI82UE 45270897 IC50 = 86 nM T48069 C36ICQ 45270898 IC50 = 19 nM T48069 C38PUJ 45271185 IC50 = 749 nM T48069 C9G6HA 45271189 IC50 = 4 nM T48069 C5KLZ9 45271190 IC50 = 4 nM T48069 C60DIT 45271191 IC50 = 20793 nM T48069 CLOB70 45271736 IC50 = 20 nM T48069 CEO73Q 45272094 IC50 = 1262 nM T48069 C4EAO2 45272095 IC50 = 286 nM T48069 C96UFP 45272096 IC50 = 1015 nM T48069 C36DGY 45272290 IC50 > 40000 nM T48069 COT0W8 45272300 IC50 = 4500 nM T48069 CE8X9I 45272611 IC50 = 90 nM T48069 CVL7R9 45272924 IC50 = 2198 nM T48069 CRC02V 45272925 IC50 = 36 nM T48069 C47LVJ 45272927 IC50 = 20 nM T48069 C1JCQ5 45272930 IC50 = 251 nM T48069 C1K2FQ 45272931 IC50 = 517 nM T48069 CY12TM 45272932 IC50 = 212 nM T48069 CC79UA 45273165 IC50 = 12600 nM T48069 CNR8G6 45273175 IC50 > 40000 nM T48069 C4UM6Y 45273507 IC50 = 170 nM T48069 CLX86A 45380509 IC50 = 23 nM T48069 CL41HJ 45380693 IC50 = 13 nM T48069 C9NCV4 45380694 IC50 = 15 nM T48069 C6SZ8A 45380791 IC50 = 46 nM T48069 CEM0V9 45380893 IC50 = 17 nM T48069 CU7Z8X 45381216 IC50 = 32 nM T48069 CWA35Y 45381330 IC50 = 5 nM T48069 C5I3OG 45381546 IC50 = 26 nM T48069 C9UF1Z 45381640 IC50 = 8 nM T48069 CP3HD2 45381723 IC50 = 60 nM T48069 C4AM7K 45381799 IC50 = 9 nM T48069 CG1QY5 45381801 IC50 = 20 nM T48069 CO4BT1 45381802 IC50 = 60 nM T48069 CT21WU 45381890 IC50 = 6 nM T48069 CWJM09 45381983 IC50 = 9 nM T48069 CZ58FY 46215814 IC50 > 10000 nM T48069 C92KBM 46229161 IC50 = 9000 nM T48069 C9Z7OT 46229173 IC50 = 63900 nM T48069 CUF3W7 46229174 IC50 = 28000 nM T48069 C6YPX1 46229187 IC50 > 100000 nM T48069 CSZX01 46229262 IC50 = 23 nM T48069 CYZV41 46231219 IC50 = 8533 nM T48069 C7J5UP 46231220 IC50 = 3198 nM T48069 CC96GZ 46231221 IC50 = 4241 nM T48069 CYT37A 46232443 IC50 > 50000 nM T48069 C48ZVW 46232555 IC50 > 50000 nM T48069 CS9B1U 46232556 IC50 = 27000 nM T48069 C7ON5A 46233287 IC50 > 10000 nM T48069 CW0P5B 46845702 IC50 = 1070 nM T48069 C7KM0E 46845704 IC50 = 1790 nM T48069 COTJ39 46863083 IC50 = 12000 nM T48069 CCBE34 46865992 IC50 = 330 nM T48069 CLS29B 46872626 IC50 > 10000 nM T48069 CF4OY7 46881850 IC50 = 81 nM T48069 C6MHP5 46881851 EC50 = 86 nM T48069 CEKX49 46881918 IC50 = 81 nM T48069 CRE96X 46885625 IC50 = 158 nM T48069 CAB87H 46886244 IC50 > 12500 nM T48069 C92HEB 46886245 IC50 > 12500 nM T48069 C5WFQ8 46886310 IC50 > 12500 nM T48069 C7S8RG 46886311 IC50 > 12500 nM T48069 CO13IV 46886312 IC50 > 12500 nM T48069 C70PZE 46886313 IC50 = 1500 nM T48069 CE8HR2 46886314 IC50 = 1300 nM T48069 CG5KO9 46886315 IC50 = 1100 nM T48069 CIFR42 46886316 IC50 = 580 nM T48069 CH5DC2 46886317 IC50 = 590 nM T48069 C2WKO4 46886318 IC50 = 450 nM T48069 CMVZ46 46886319 IC50 = 130 nM T48069 CW19TR 46886320 IC50 = 3800 nM T48069 CJR01I 46886321 IC50 = 200 nM T48069 CL50ZE 46886322 IC50 = 100 nM T48069 C2O8RZ 46886323 IC50 = 140 nM T48069 CN30BX 46886324 IC50 = 81 nM T48069 CC7MG8 46886325 IC50 = 41 nM T48069 C0L1EW 46886326 IC50 = 46 nM T48069 C3T6YO 46886327 IC50 = 27 nM T48069 CL5R0D 46888599 IC50 = 2960 nM T48069 C3IE0X 46888601 IC50 = 990 nM T48069 C1A0XQ 46888603 IC50 = 3210 nM T48069 CB5YQ1 46888635 IC50 = 2250 nM T48069 C6YC4O 46888663 IC50 = 2360 nM T48069 C0AUT8 46888665 IC50 = 1780 nM T48069 CAZT96 46888666 IC50 > 50000 nM T48069 CS4U3P 46888668 IC50 = 980 nM T48069 CASV10 46888710 IC50 = 2860 nM T48069 CY2TV5 46888712 IC50 = 5150 nM T48069 CX5AL6 46888740 IC50 = 1330 nM T48069 CSWE93 46888742 IC50 = 10610 nM T48069 C7YN9L 46927873 IC50 = 3500 nM T48069 CR1ZT4 46927874 IC50 = 5200 nM T48069 CT1DF3 46927875 IC50 = 5600 nM T48069 C60GAV 46929544 IC50 > 8000 nM T48069 CP34VL 46929748 IC50 > 1000 nM T48069 CJ2E9Q 46929857 IC50 > 25000 nM T48069 CHSF07 49806372 IC50 > 1000 nM T48069 C5ME3S 49806721 IC50 > 50000 nM T48069 C9L3XR 49838879 IC50 > 50000 nM T48069 CB74UR 49864985 IC50 = 190 nM T48069 CCBX17 49864986 IC50 = 32 nM T48069 C82HPG 49865038 IC50 = 5.3 nM T48069 C5RQ7C 50908680 Ki = 110 nM T48069 CD2K4R 50908681 Ki = 150 nM T48069 C4DH0A 50938549 IC50 = 6 nM T48069 CS9G6E 50997096 IC50 > 10000 nM T48069 CAZQ43 51003133 IC50 > 1000 nM T48069 CO7U5C 51355838 IC50 = 9.4 nM T48069 CIXL91 51355841 IC50 = 21 nM T48069 CUR7Z0 52918127 IC50 = 7 nM T48069 CXA03W 52920796 IC50 > 100 nM T48069 CEQN27 52936621 Ki > 1000 nM T48069 CM24LF 52938983 IC50 = 51.62 nM T48069 C8LG3X 52941007 IC50 > 30000 nM T48069 CI4Q9G 52941251 IC50 = 6700 nM T48069 CO6LK0 52941271 IC50 = 27100 nM T48069 CUK07B 52941277 IC50 > 30000 nM T48069 C2ZTN3 52941514 IC50 = 7.5 nM T48069 C8XN0Y 52941515 IC50 = 348 nM T48069 CG9E4A 52942446 Ki = 580 nM T48069 CJN4X2 52942639 IC50 > 30000 nM T48069 C23VML 52942746 IC50 = 415 nM T48069 CT37AH 52942747 IC50 = 22 nM T48069 C41KCI 52942861 IC50 = 179 nM T48069 C8SJ2Q 52942862 Ki > 1000000 nM T48069 CA51LB 52943781 IC50 = 107.15 nM T48069 CUM65L 52943909 IC50 = 12500 nM T48069 C8V2TG 52943910 IC50 = 20500 nM T48069 CWX4M7 52943942 IC50 > 30000 nM T48069 CLO46D 52944812 Ki = 2110 nM T48069 C26OFX 52944836 IC50 > 30000 nM T48069 CZR27V 52944899 IC50 = 15400 nM T48069 CU3LH6 52944953 IC50 = 21100 nM T48069 CAT41H 52944991 IC50 = 21400 nM T48069 C61WJR 52945091 IC50 = 6500 nM T48069 C6FIA5 52945092 IC50 = 24700 nM T48069 CW09EM 52945447 IC50 = 180 nM T48069 CNV67T 52945448 IC50 = 2450 nM T48069 CMK4V1 52945862 IC50 > 30000 nM T48069 CD5YH8 52946371 IC50 = 45.1 nM T48069 CGA62C 52946372 IC50 = 283 nM T48069 C09UQW 52946470 IC50 = 4.1 nM T48069 CIC58E 52946503 IC50 = 42 nM T48069 C30RAL 52946684 IC50 = 1300 nM T48069 C8WK7M 52947405 IC50 = 14900 nM T48069 CW3A6V 52947411 IC50 > 30000 nM T48069 CRN80K 52947412 IC50 > 30000 nM T48069 CQ0V4I 52947602 IC50 = 72.4 nM T48069 CYQ4L3 52947603 IC50 = 49 nM T48069 C93VNZ 52947604 IC50 = 194.98 nM T48069 C5ZT3P 52947609 IC50 > 30000 nM T48069 CYBQ53 52947703 IC50 = 19300 nM T48069 CI6GX2 52948511 Ki = 570 nM T48069 C09KRB 52948552 IC50 = 28100 nM T48069 CC7D8Y 52948708 IC50 > 30000 nM T48069 CTY9Z8 52948817 IC50 = 125.89 nM T48069 CWA74O 52949707 Ki = 370 nM T48069 C4XMC6 52949728 IC50 = 8800 nM T48069 C1LVR8 52949876 IC50 > 30000 nM T48069 CPAM54 52950015 IC50 = 94 nM T48069 CO9QW4 52950016 IC50 = 112.2 nM T48069 C0M2SG 52950017 IC50 = 115 nM T48069 C6OTY5 53251320 IC50 > 30000 nM T48069 C09SDH 53257410 IC50 > 10000 nM T48069 CVL9H8 53316637 IC50 = 6 nM T48069 CR5Z6P 53316638 IC50 = 5 nM T48069 C0NT5S 53316639 IC50 = 20 nM T48069 CE8OY2 53317913 IC50 > 100 nM T48069 CJ2D3F 53319267 IC50 = 17 nM T48069 C8UVK2 53319268 IC50 = 8 nM T48069 C24OPK 53319269 IC50 = 2 nM T48069 C5DUO3 53319892 IC50 = 8 nM T48069 CNQF53 53320577 IC50 = 285 nM T48069 C24TVU 53321197 IC50 = 150 nM T48069 C5B2LC 53321198 IC50 = 26 nM T48069 CIJ3R9 53321874 IC50 = 4 nM T48069 CL7OG4 53323210 IC50 = 5 nM T48069 CSL19U 53323211 IC50 = 5 nM T48069 CH3TR6 53323212 IC50 = 5 nM T48069 C6TQD2 53323213 IC50 = 8 nM T48069 C2W9OA 53324451 IC50 > 10000 nM T48069 C3X9HS 53324563 IC50 = 21 nM T48069 C85XCF 53324564 IC50 = 14 nM T48069 CEK97L 53325637 IC50 = 25 nM T48069 C0VS2G 53326809 IC50 = 27 nM T48069 C5EOS8 53328013 IC50 = 670 nM T48069 COJ3C2 53328118 IC50 = 82000 nM T48069 CNET81 53328119 IC50 = 54000 nM T48069 CVC5T4 53328120 IC50 = 4400 nM T48069 C9PR3G 53328121 IC50 = 4100 nM T48069 CG0I5B 53328122 IC50 = 16000 nM T48069 C8WJC1 53328317 IC50 = 4000 nM T48069 C4R1OF 53328318 IC50 = 91000 nM T48069 C2YC0W 53328319 IC50 = 4900 nM T48069 CJIE57 53328320 IC50 = 12000 nM T48069 C6XQ3O 53328321 IC50 = 31000 nM T48069 CKQA18 53328322 IC50 = 4900 nM T48069 CHC90P 53328509 IC50 = 810 nM T48069 CNG20E 53328510 IC50 = 990 nM T48069 CA2N6W 53328511 IC50 = 680 nM T48069 C72RMJ 53328512 IC50 = 3300 nM T48069 C92VPI 53330628 IC50 > 100000 nM T48069 CI23LK 53330629 IC50 > 100000 nM T48069 CEO7M1 53330630 IC50 > 100000 nM T48069 CNPM14 53341082 IC50 > 3000 nM T48069 C8ZRE3 53356518 IC50 = 17910 nM T48069 CM7P3W 53357328 IC50 = 1000 nM T48069 CBK9Q6 53357848 IC50 > 10000 nM T48069 CK52GI 53380818 IC50 = 17 nM T48069 C8NA4L 53384644 IC50 > 30000 nM T48069 CVG90B 53389651 IC50 > 10000 nM T48069 C5VG9P 53495177 IC50 = 116 nM T48069 CVC7Z5 54580422 IC50 = 4706 nM T48069 CE8R0Y 54581423 IC50 = 1089 nM T48069 CON48Z 54581424 IC50 = 995 nM T48069 CKJ76V 54581425 IC50 = 34 nM T48069 C61AXC 54581467 IC50 = 48 nM T48069 C23PAV 54582434 IC50 = 2950 nM T48069 C5ZLJ4 54582435 IC50 = 574 nM T48069 CT19GU 54582436 IC50 = 47 nM T48069 CE5MH6 54583413 IC50 > 10000 nM T48069 C5C6QV 54583414 IC50 > 10000 nM T48069 CXM14L 54583415 IC50 = 4501 nM T48069 C2B6SJ 54583448 IC50 = 34 nM T48069 COA58F 54584367 IC50 > 10000 nM T48069 CMLB37 54584368 IC50 = 1241 nM T48069 CD5TK9 54584369 IC50 = 453 nM T48069 CE9O1Z 54585334 IC50 > 10000 nM T48069 C3E2OK 54585335 IC50 > 10000 nM T48069 CF50GC 54585372 IC50 = 2.2 nM T48069 CC78IN 54585373 IC50 = 933 nM T48069 CS13HO 54586287 IC50 = 117 nM T48069 CA3SP2 54586288 IC50 > 10000 nM T48069 CRY0W5 54586289 IC50 = 1061 nM T48069 C0YH6B 54586290 IC50 = 784 nM T48069 C6XH4I 54586291 IC50 = 703 nM T48069 CYT4P9 54586292 IC50 = 202 nM T48069 CSW58D 54586329 IC50 = 9219 nM T48069 CPV4T0 54587318 IC50 = 2897 nM T48069 C4EAG8 54587319 IC50 = 1851 nM T48069 C3WOR4 54587320 IC50 = 1052 nM T48069 CA85KR 54587364 IC50 = 36 nM T48069 CT71UH 54596950 IC50 = 798 nM T48069 C2F6DB 54596952 IC50 = 4230 nM T48069 CE1ZK6 54759168 IC50 > 10000 nM T48069 C1XS2J 54760383 IC50 > 10000 nM T48069 C9ZFS1 54764923 IC50 = 3160 nM T48069 CRH20S 56596558 IC50 = 4610 nM T48069 CM8JX1 56604907 IC50 = 10 nM T48069 CZBP85 56659843 IC50 = 450 nM T48069 C1ILG0 56659844 IC50 = 47 nM T48069 COH8L9 56659845 IC50 = 13 nM T48069 CGJ0C9 56663313 IC50 = 10 nM T48069 C8OJ7L 56663314 IC50 = 10 nM T48069 CL8IE7 56663315 IC50 = 270 nM T48069 C9T2JQ 56663564 IC50 = 41 nM T48069 C1KDU3 56663565 IC50 = 40 nM T48069 CO1E6D 56663566 IC50 = 17 nM T48069 CED2I5 56663567 IC50 = 51 nM T48069 CS5XV2 56666509 IC50 = 92 nM T48069 CMH52U 56666742 IC50 = 35 nM T48069 CUL0F4 56667010 IC50 = 39 nM T48069 C9G1FY 56667011 IC50 = 8 nM T48069 CA6K8E 56667012 IC50 = 47 nM T48069 C2HXG3 56667013 IC50 = 1060 nM T48069 C0HA7C 56670167 IC50 = 270 nM T48069 C1OT4M 56670168 IC50 = 13 nM T48069 CT7YZ8 56670169 IC50 = 140 nM T48069 CR28XB 56670170 IC50 = 9 nM T48069 CE14PX 56670172 IC50 = 53 nM T48069 C76KFA 56670457 IC50 = 18 nM T48069 C0I6AP 56670458 IC50 = 4 nM T48069 C9Y8PV 56670459 IC50 = 45 nM T48069 C5E7OB 56670460 IC50 = 11 nM T48069 CCPY59 56670461 IC50 = 6 nM T48069 CYJF34 56673688 IC50 = 89 nM T48069 CR0O6E 56673689 IC50 = 190 nM T48069 C8QCI3 56673690 IC50 = 49 nM T48069 CK5HP1 56673946 IC50 = 33 nM T48069 C2D4JW 56673947 IC50 = 5 nM T48069 CPU13M 56673948 IC50 = 31 nM T48069 CK0ZR4 56677003 IC50 = 40 nM T48069 CTW73X 56677275 IC50 = 2 nM T48069 CHG64Z 56677276 IC50 = 4 nM T48069 CQJ9N1 56680334 IC50 = 3 nM T48069 CR80OL 56680335 IC50 = 35 nM T48069 C1AOI5 56680336 IC50 = 11 nM T48069 CTS0D4 56680337 IC50 = 60 nM T48069 C67GMA 56680575 IC50 = 83 nM T48069 C2P3RA 56683651 IC50 = 15 nM T48069 CQP42U 56683652 IC50 = 8 nM T48069 CGTH28 56683653 IC50 = 210 nM T48069 C81IHQ 56683654 IC50 = 10 nM T48069 CHFC24 56683655 IC50 = 55 nM T48069 C0CEU6 56683656 IC50 = 22 nM T48069 CWBF48 56683908 IC50 = 13 nM T48069 CF5JV6 56966833 IC50 = 20.3 nM T48069 C1WJT2 56966906 IC50 = 59.5 nM T48069 C26MCX 56966977 IC50 = 98.1 nM T48069 CX34KP 56966978 IC50 = 8.2 nM T48069 CDS06V 56973548 IC50 = 6309.57 nM T48069 CUAV97 56973549 IC50 = 19952.62 nM T48069 CI0K7Y 56973550 IC50 = 6309.57 nM T48069 CPHX64 57325478 IC50 > 50000 nM T48069 CQ9BW4 57325479 IC50 > 50000 nM T48069 C56XYJ 57325607 IC50 = 1870 nM T48069 C09DJP 57325609 IC50 = 503 nM T48069 C95OSR 57325611 IC50 > 25000 nM T48069 CJ93CQ 57325613 IC50 = 8890 nM T48069 CB6UG1 57325697 IC50 > 25000 nM T48069 CZUV79 57325700 IC50 > 25000 nM T48069 CKQF98 57325702 IC50 = 2770 nM T48069 CGN9R7 57326499 IC50 > 25000 nM T48069 C1M2SJ 57326501 IC50 > 25000 nM T48069 C7HSP3 57326503 IC50 > 25000 nM T48069 C06SPM 57326505 IC50 > 25000 nM T48069 CIRD14 57326601 IC50 > 25000 nM T48069 CUCT15 57326603 IC50 > 25000 nM T48069 CY5AW1 57326605 IC50 = 9022 nM T48069 CY6JT2 57326607 IC50 > 25000 nM T48069 C8X0KC 57326609 IC50 > 25000 nM T48069 CNW2D1 57326700 IC50 > 25000 nM T48069 CSV93R 57326702 IC50 > 25000 nM T48069 C0QU2R 57326704 IC50 > 25000 nM T48069 CML95J 57326706 IC50 = 2930 nM T48069 CF65OP 57326708 IC50 = 6590 nM T48069 C5K1TC 57326800 IC50 = 6120 nM T48069 C1Y9WO 57326802 IC50 > 25000 nM T48069 C5P8CS 57326804 IC50 = 6390 nM T48069 CH92NG 57326806 IC50 = 4100 nM T48069 CIE2N9 57326900 IC50 = 10540 nM T48069 CT4HO0 57326902 IC50 > 25000 nM T48069 C6DWX9 57326904 IC50 = 8320 nM T48069 C86FYD 57326906 IC50 = 722 nM T48069 CU8L3K 57326995 IC50 = 7080 nM T48069 C4AI8K 57326997 IC50 = 364 nM T48069 CH87XA 57398439 IC50 = 5 nM T48069 C0UDY9 57401151 IC50 > 30000 nM T48069 CJK85L 57403635 IC50 = 6 nM T48069 C31PRG 57403636 IC50 = 10 nM T48069 CZSM95 57412684 IC50 > 10000 nM T48069 C8P6RD 57505528 IC50 > 10000 nM T48069 CVK0G4 58056356 IC50 > 50000 nM T48069 C7HPC2 58268648 Ki = 557 nM T48069 C6BPR2 58985201 IC50 > 30000 nM T48069 CBWJ84 59291203 IC50 = 20 nM T48069 CT3EW2 59292007 IC50 > 1000 nM T48069 C24BEZ 59577331 IC50 = 364 nM T48069 CT3J2N 59577341 IC50 = 244 nM T48069 CIB62O 59577356 IC50 = 391 nM T48069 C75VNB 59577361 IC50 = 903 nM T48069 C7QY2B 59577365 IC50 = 181 nM T48069 C1E3OI 59598370 Ki = 730 nM T48069 CQ2UE7 59598391 Ki = 637 nM T48069 C5AEN1 59598393 Ki = 217 nM T48069 CUA1F5 59598396 Ki = 1330 nM T48069 C0O6ZX 59598404 Ki = 575 nM T48069 CBMH78 59598415 Ki = 2890 nM T48069 CYNP39 59598421 Ki = 864 nM T48069 CU1ER8 59598432 Ki = 27 nM T48069 C0L5DN 59598437 Ki = 190 nM T48069 CKVB01 59598456 Ki = 250 nM T48069 CXJ63M 59603829 IC50 > 100000 nM T48069 CQEU96 59603842 IC50 = 2800 nM T48069 CCX2Q5 59864465 Ki = 618 nM T48069 C1MR8Q 60097495 IC50 > 1000 nM T48069 COM48T 60154284 IC50 = 3981.07 nM T48069 CB7KE0 60154285 IC50 = 6309.57 nM T48069 CO75BK 60154286 IC50 = 10000 nM T48069 CEF48W 60154326 IC50 = 398.11 nM T48069 C2Y7JC 60154327 IC50 = 7943.28 nM T48069 COU2B3 60154328 IC50 = 12589.25 nM T48069 CKM5E6 60154329 IC50 = 31622.78 nM T48069 CVE49A 60154330 IC50 = 15848.93 nM T48069 C3BMS1 60154331 IC50 = 12589.25 nM T48069 CBU4I5 60154332 IC50 = 6309.57 nM T48069 C03CFA 60154333 IC50 = 3981.07 nM T48069 CLK0O6 60154334 IC50 = 12589.25 nM T48069 C34QJR 60154335 IC50 = 15848.93 nM T48069 CXO1I8 60154336 IC50 = 50118.72 nM T48069 CNZX63 60154337 IC50 = 10000 nM T48069 C3I4KJ 60154338 IC50 = 7943.28 nM T48069 CRB5D8 60154339 IC50 = 39810.72 nM T48069 CYI9F7 60154340 IC50 = 3162.28 nM T48069 CLY46E 60154341 IC50 = 100 nM T48069 CNS3Y1 60154342 IC50 = 1584.89 nM T48069 C7CS4I 60154343 IC50 = 398.11 nM T48069 C46LSW 60154344 IC50 = 12589.25 nM T48069 CR60YI 60154345 IC50 = 100000 nM T48069 C0NC7M 66547682 IC50 = 47 nM T48069 CRU40E 67034649 IC50 = 490 nM T48069 C1GQ6Z 67034810 IC50 = 33 nM T48069 CDE5H6 67035079 IC50 = 47 nM T48069 C1HSE0 67035086 IC50 = 420 nM T48069 CWI6K5 67035106 IC50 = 14 nM T48069 CC1WL3 67035462 IC50 = 130 nM T48069 C42MZP 67035535 IC50 = 80 nM T48069 C38RGB 67035556 IC50 = 80 nM T48069 CV3HW2 67035568 IC50 = 9 nM T48069 CXU54K 67035992 IC50 = 60 nM T48069 C37NKO 67129970 IC50 > 10000 nM T48069 CK80LJ 67130050 IC50 > 10000 nM T48069 CV63UL 67240318 IC50 > 10000 nM T48069 CDMS72 67980571 IC50 = 80 nM T48069 CEV60X 68156947 IC50 = 1.9 nM T48069 C59RQC 68165302 IC50 = 45.1 nM T48069 CL97JB 68165311 IC50 = 51.4 nM T48069 CM1ZC3 68165315 IC50 = 17.4 nM T48069 CET2P8 68165322 IC50 = 43.3 nM T48069 C61QGN 68165327 IC50 = 42.7 nM T48069 CFRK82 68165328 IC50 = 0.4 nM T48069 CLH97K 68165338 IC50 = 143 nM T48069 C7Y8KG 68165350 IC50 = 26.9 nM T48069 C2AX3V 68165354 IC50 = 38.8 nM T48069 C2B3TL 68165357 IC50 = 128 nM T48069 C81YOZ 68165362 IC50 = 86.5 nM T48069 CLGN08 68165375 IC50 = 0.11 nM T48069 C82RIW 68165380 IC50 = 103 nM T48069 CH5Y2P 68165382 IC50 = 77.5 nM T48069 C3H5XQ 68165389 IC50 = 31.6 nM T48069 C0WFX2 68165395 IC50 = 0.47 nM T48069 C0G7QF 68165398 IC50 = 203 nM T48069 CNK7S3 68165399 IC50 = 32.5 nM T48069 C78BZG 68165403 IC50 = 20.3 nM T48069 CZ1Q8W 68165412 IC50 = 22.1 nM T48069 CYD2V8 68165414 IC50 = 27 nM T48069 CVGJ74 68165424 IC50 = 6.2 nM T48069 CN27QC 68165467 IC50 = 434 nM T48069 CO2LF9 68166178 IC50 = 81.5 nM T48069 CR1U7L 68166323 IC50 = 100 nM T48069 C4VQJ8 68166330 IC50 = 125 nM T48069 C8I7GC 68293638 IC50 = 13 nM T48069 CD56XK 68293660 IC50 = 15 nM T48069 CS98LK 68293683 IC50 = 7.3 nM T48069 CVJX68 68293694 IC50 = 14 nM T48069 CE6B8L 68293755 IC50 = 7.8 nM T48069 C4U2HY 68293779 IC50 = 4.3 nM T48069 C8Q6LH 68293853 IC50 = 2.8 nM T48069 C7GRV2 68755406 IC50 > 10000 nM T48069 C5DGR9 69036886 IC50 = 2137 nM T48069 CUEO45 70681644 Ki = 149 nM T48069 C59QUO 70683775 Ki = 93.6 nM T48069 C3RQ0D 70683776 Ki = 3100 nM T48069 C3O4UL 70688040 Ki = 948 nM T48069 C4CY2F 70690067 Ki = 146 nM T48069 CL0F7V 70690072 Ki = 708 nM T48069 C7I6QX 70690073 Ki = 1660 nM T48069 C3OVZ0 70692216 Ki = 233 nM T48069 CLZ65T 70692217 Ki = 680 nM T48069 CEBO91 71452977 IC50 > 10000 nM T48069 CKT60L 71455860 Ki > 1800 nM T48069 CCR8J9 71496459 IC50 = 1600 nM T48069 C8V4GQ 71496460 IC50 = 263000 nM T48069 CRX81Q 71575642 IC50 > 10000 nM T48069 CZ31PU 71583657 IC50 > 10000 nM T48069 CLMU95 71762923 IC50 = 0.7 nM T48069 CGZ7X8 71762924 IC50 = 0.6 nM T48069 C3G4IT 71762925 IC50 = 10 nM T48069 CK9D0J 71762926 IC50 = 23 nM T48069 CQL13N 71763139 IC50 = 4 nM T48069 CO2NQ0 71763140 IC50 = 5 nM T48069 CHA3X9 71763141 IC50 = 10 nM T48069 C5HP1X 71763142 IC50 = 8 nM T48069 C43COT 71763143 IC50 = 16 nM T48069 CK7LW6 71763375 IC50 = 24 nM T48069 CH5YW8 71763376 IC50 = 29 nM T48069 CD7Q6P 71763377 IC50 = 195 nM T48069 CR8J2G 71763378 IC50 = 9 nM T48069 CZ9P5A 71763605 IC50 = 9 nM T48069 CZ3A1G 71763606 IC50 = 26 nM T48069 C5FX7O 71763607 IC50 = 72 nM T48069 CBY80T 72716071 IC50 = 779 nM T48069 C60TUV 72737208 IC50 > 10000 nM T48069 CJ3WA6 72737404 IC50 > 10000 nM T48069 CG8RI0 73292361 IC50 = 2 nM T48069 CBQ72N 73292545 IC50 = 813 nM T48069 CQV1P0 73294507 IC50 = 4 nM T48069 CVNW01 73386831 IC50 > 1000 nM T48069 C3UC9H 73891099 IC50 = 70 nM T48069 C40WYO 76286188 IC50 = 30 nM T48069 CDQ87J 76286189 IC50 = 1186 nM T48069 CON96X 76286190 IC50 = 2081 nM T48069 C4NIS8 76286191 IC50 = 235 nM T48069 CGMQ70 76286192 IC50 = 1107 nM T48069 CA2XL0 76286346 IC50 = 98 nM T48069 CNX63K 76286347 IC50 = 265 nM T48069 CLHO60 76286348 IC50 = 207 nM T48069 C9CS5E 76286349 IC50 = 129 nM T48069 C85SPH 76286350 IC50 = 270 nM T48069 CON1Y6 76286351 IC50 = 395 nM T48069 CZU79O 76286494 IC50 = 374 nM T48069 CV8QX0 76310169 IC50 = 2040 nM T48069 CA5L4W 76324771 IC50 = 3500 nM T48069 C9GO0P 76328313 IC50 = 560 nM T48069 C39FTZ 76335685 IC50 = 3310 nM T48069 CV0P3A 78357783 IC50 = 7000 nM T48069 CCJ43A 86302281 IC50 > 10000 nM T48069 CB5NJ4 86302541 IC50 > 10000 nM T48069 CPG3A5 86302574 IC50 > 30000 nM T48069 C9NTP1 86677234 IC50 = 7 nM T48069 C5YX8T 86677253 IC50 = 196000 nM T48069 CCX1U5 86677265 IC50 = 40000 nM T48069 CZQ1F7 86677270 IC50 = 38000 nM T48069 CLJ36F 86705466 IC50 = 31 nM T48069 C1HW4B 89735655 IC50 > 100000 nM T48069 CH58TV 89773144 IC50 = 117 nM T48069 CSX63K 89773146 IC50 = 8.7 nM T48069 CTV2C7 89774514 IC50 = 47.3 nM T48069 CX29IY 90655145 IC50 > 10000 nM T48069 CP34KC 90664681 IC50 = 2760 nM T48069 CK3IS4 90664930 IC50 = 2800 nM T48069 CB5GU0 91668530 IC50 = 3300 nM T48069 CAU45T 91971978 IC50 > 30000 nM T48069 C05NTY 101884761 IC50 = 26 nM T48069 CWM71R 101884762 IC50 = 6 nM T48069 CU6P5O 117929138 IC50 > 1000 nM T48069 C3HKM8 117929389 IC50 = 10 nM T48069 CI1B0H 117929423 IC50 > 1000 nM T48069 CQIP89 117929456 IC50 = 58 nM T48069 C9K0CN 117929460 IC50 = 35 nM T48069 CL9G2E 117929486 IC50 > 1000 nM T48069 CN0EF8 117929515 IC50 = 20 nM T48069 CYTS68 117929557 IC50 > 1000 nM T48069 C4PYW5 117929716 IC50 = 786 nM T48069 C5BNK4 117929727 IC50 = 2800 nM T48069 CM1U4W 117929761 IC50 = 1190 nM T48069 C2S9XV 117930041 IC50 = 1500 nM T48069 C3KLI5 118723185 IC50 > 100000 nM T48069 CAP45I 118731838 IC50 > 1000 nM T48069 CMB2F4 118731839 IC50 = 32 nM T48069 CUWH39 118731840 IC50 = 90 nM T48069 CDJ2R5 118731841 IC50 = 184 nM T48069 C1X4BM 118731842 IC50 = 203 nM T48069 CO7T1R 118731843 IC50 = 124 nM T48069 CR4AY0 118731844 IC50 = 41 nM T48069 CLWK87 118731845 IC50 = 267 nM T48069 C4SL8J 118731846 IC50 = 149 nM T48069 C4QMY0 118731847 IC50 = 97 nM T48069 CYMS03 118731848 IC50 = 442 nM T48069 CX9M3K 118731850 IC50 = 2000 nM T48069 CXC4F5 118731851 IC50 = 970 nM T48069 CYKU80 118731852 IC50 = 251 nM T48069 C96CNP 118731853 IC50 = 300 nM T48069 C18JON 118731854 IC50 = 568 nM T48069 C62ZUO 118731855 IC50 = 108 nM T48069 CP27TX 118735321 IC50 = 2409 nM T48069 CJH0M1 118735322 IC50 > 100000 nM T48069 CA7Z4X 118735323 IC50 = 34125 nM T48069 C76XKT 118735324 IC50 = 40515 nM T48069 CI26FD 118735325 IC50 > 100000 nM T48069 CU8T1C 118735326 IC50 = 965 nM T48069 C1PDE5 118735327 IC50 = 1489 nM T48069 CQ0GS4 118735328 IC50 = 72 nM T48069 C3KLT1 118735329 IC50 = 51 nM T48069 C1RAP6 118735330 IC50 = 3174 nM T48069 CQ45PF 118735331 IC50 = 30 nM T48069 C56MYE 118735332 IC50 = 67727 nM T48069 CP26VF 118735333 IC50 > 100000 nM T48069 CSR3N8 118735334 IC50 > 10000 nM T48069 C3TS7H 118735335 IC50 > 29000 nM T48069 C4DQ5K 118735336 IC50 = 46942 nM T48069 C4DQX9 118735337 IC50 > 100000 nM T48069 CBY4K3 118735338 IC50 > 100000 nM T48069 C5CK7W 118735339 IC50 = 7992 nM T48069 CV06MA 122177111 IC50 = 14 nM T48069 C2DH7M 122177112 IC50 = 38 nM T48069 CL8GC2 122177113 IC50 = 9 nM T48069 C08KEM 122179540 IC50 = 4000 nM T48069 CG0RP7 122179547 IC50 = 5100 nM T48069 C1A0SQ 122179548 IC50 = 5400 nM T48069 C4X7SD 122192466 IC50 > 10000 nM T48069 COF75Z 126970673 IC50 = 48 nM T48069 C8KXV1 127025843 IC50 > 1000 nM T48069 C5SAZ7 127030054 IC50 = 260 nM T48069 CL0YQ5 127030360 IC50 = 840 nM T48069 CV38CP 127031035 IC50 = 160 nM T48069 CWTM38 127031036 IC50 = 370 nM T48069 CWE52N 127031915 IC50 = 1900 nM T48069 C7FW5G 127031916 IC50 = 110 nM T48069 CVG52X 127033379 IC50 = 200 nM T48069 CCZU26 127033936 IC50 = 3700 nM T48069 CH0UI6 127033937 IC50 = 550 nM T48069 C86SBK 127033954 IC50 = 1291 nM T48069 CJCR47 127033955 IC50 = 5602 nM T48069 CPJL35 127034194 IC50 = 2000 nM T48069 CZJG87 127034195 IC50 = 7900 nM T48069 C9UV5Q 127034463 IC50 = 630 nM T48069 CH05NE 127034464 IC50 = 310 nM T48069 CKS28E 127034802 IC50 = 27.8 nM T48069 CKX40V 127037812 IC50 > 10000 nM T48069 C70RUP 127038480 IC50 > 10000 nM T48069 C3WCN8 127041777 IC50 > 10000 nM T48069 CHK16Q 127045929 IC50 > 1000 nM T48069 CY3J0C 127047591 IC50 > 1000 nM T48069 CSEJ41 127048207 IC50 = 136 nM T48069 CDK3C6 127049147 IC50 = 51.6 nM T48069 C2MF9I 127049148 IC50 = 1.4 nM T48069 CV1E5D 127049149 IC50 = 6.17 nM T48069 C07TZN 127049440 IC50 = 1.93 nM T48069 C2FE1A 127049463 IC50 = 1.33 nM T48069 C7ODG2 127049464 IC50 = 36.1 nM T48069 C7A4OJ 127049465 IC50 = 0.76 nM T48069 C7D5QM 127049475 IC50 = 12 nM T48069 C3V9MD 127049476 IC50 = 10 nM T48069 CS6C8O 127050851 IC50 = 14 nM T48069 C1HAU4 127050852 IC50 = 29 nM T48069 CHVU86 127050853 IC50 = 15 nM T48069 CWDX26 127050854 IC50 = 31 nM T48069 C7DU0N 127050855 IC50 = 39 nM T48069 CLX8S5 127050856 IC50 = 9 nM T48069 CH46LU 127051126 IC50 = 6 nM T48069 C39WXP 127051127 IC50 = 8 nM T48069 C5J3KY 127051128 IC50 = 5 nM T48069 C7E4QP 127051129 IC50 = 6 nM T48069 CDJQ32 127051599 IC50 = 42 nM T48069 C2ISZ9 127051600 IC50 = 76 nM T48069 C61GFX 127051601 IC50 = 35 nM T48069 CFQ2X7 127051618 IC50 = 24 nM T48069 C4DSF7 127051619 IC50 = 49 nM T48069 C8JMN0 127051620 IC50 = 49 nM T48069 CTZK49 127051621 IC50 = 6 nM T48069 C7PZM3 127051622 IC50 = 8 nM T48069 CZO5C7 127052225 IC50 = 12 nM T48069 COX90Y 127052226 IC50 = 29 nM T48069 CHQJ02 127052979 IC50 = 51.6 nM T48069 CUO0C5 132156633 IC50 > 10000 nM T48069 C4Q5LF 132471857 IC50 > 30000 nM T48069 CERS64 132937256 IC50 > 30000 nM T48069 CN35SO 134146628 IC50 > 1000 nM T48069 CYL5V1 134694986 IC50 > 30000 nM T48069 CQ54JK 135410197 IC50 = 72800 nM T48069 CZJ62H 135423375 IC50 = 61 nM T48069 C80RLK 135424490 IC50 = 590 nM T48069 CAJ2C0 135448904 IC50 = 16 nM T48069 CM95TC 135452916 IC50 = 300 nM T48069 CO0RV2 135454939 IC50 = 160 nM T48069 CUB5X7 135469646 IC50 = 140 nM T48069 CLSZ84 135497093 IC50 = 3310 nM T48069 CTJ48K 135524085 IC50 = 6400 nM T48069 CUT1W7 135524168 IC50 > 10000 nM T48069 CRT3X6 135524445 IC50 = 2900 nM T48069 CC3V9D 135529500 IC50 > 25000 nM T48069 C3RX6B 135530418 IC50 = 390 nM T48069 CSP0N8 135530495 IC50 = 190 nM T48069 CVG1B3 135532904 IC50 = 540 nM T48069 C2MAC7 135536640 IC50 > 100000 nM T48069 C95XVI 135542937 IC50 = 720 nM T48069 C7YA9M 135553232 IC50 = 18 nM T48069 C15VPC 135553240 IC50 = 38 nM T48069 CTB8U4 135553266 IC50 = 180 nM T48069 CL9Q1F 135553267 IC50 = 2500 nM T48069 C6W3AL 135553268 IC50 = 1300 nM T48069 C53HFP 135553269 IC50 = 270 nM T48069 C5Y6IB 135553271 IC50 = 550 nM T48069 CS5J2N 135553279 IC50 = 1640 nM T48069 CTY9F2 135553383 IC50 = 800 nM T48069 CY4D8I 135566504 Ki = 990.9 nM T48069 CS0Y1X 135611169 IC50 = 290 nM T48069 CJU23T 135681572 IC50 = 1200 nM T48069 CQ64XU 135681577 IC50 = 180 nM T48069 C3BN2K 135681579 IC50 = 2500 nM T48069 CZX62Q 135681587 IC50 = 3000 nM T48069 CN1T7U 135681590 IC50 = 93 nM T48069 CJ4C1Y 135681596 IC50 = 770 nM T48069 CJZ39U 135681612 IC50 = 180 nM T48069 C5DKL0 135681672 IC50 = 2100 nM T48069 CDL97B 135681674 IC50 = 14000 nM T48069 CU6CS1 135681699 IC50 > 25000 nM T48069 CNPW48 135681721 IC50 = 780 nM T48069 CIZE46 135681727 IC50 = 350 nM T48069 C3EKM9 135681730 IC50 = 170 nM T48069 C9KAC6 135681742 IC50 = 520 nM T48069 CG2W0I 135681763 IC50 = 520 nM T48069 CYJ30L 135681778 IC50 = 430 nM T48069 CAL5Y3 135681791 IC50 = 3000 nM T48069 COQZ51 135681794 IC50 = 5300 nM T48069 CR25XH 135681808 IC50 = 1590 nM T48069 C7C5VZ 135681810 IC50 = 530 nM T48069 CYV2J5 135681820 IC50 = 250 nM T48069 CI73WC 135681822 IC50 = 340 nM T48069 CMN19V 135681825 IC50 = 3050 nM T48069 COQB90 135681826 IC50 > 25000 nM T48069 C9UGN1 135681832 IC50 = 68 nM T48069 C62NOS 135681833 IC50 = 54 nM T48069 C3D0CJ 135681834 IC50 = 140 nM T48069 CIG3R9 135681875 IC50 = 46 nM T48069 CD2WU5 135681903 IC50 = 3630 nM T48069 C73SIW 135681935 IC50 = 1270 nM T48069 CJV72X 135779792 IC50 = 140 nM T48069 CAH27Z 135858938 IC50 = 169 nM T48069 CC9AU4 135869565 IC50 = 120 nM T48069 CQSV28 135875708 IC50 = 22 nM T48069 CF16XL 135875709 IC50 = 18 nM T48069 CL35XZ 135875710 IC50 = 31 nM T48069 C56WCS 135875711 IC50 = 23 nM T48069 C37BGJ 135875712 IC50 = 20 nM T48069 C9B5PC 135875713 IC50 = 26 nM T48069 CACB27 135875714 IC50 = 25 nM T48069 CKN2G0 135875715 IC50 = 18 nM T48069 CU5VY1 135922386 IC50 = 45 nM T48069 CG3UZ1 135927974 Ki > 1000 nM T48069 CIPA79 135937899 IC50 > 10000 nM T48069 CCIJ86 135960711 IC50 = 29 nM T48069 C6GS3B 135960712 IC50 = 220 nM T48069 CI9UP7 135960713 IC50 = 150 nM T48069 C4RY9Q 135960714 IC50 = 45 nM T48069 CWAH57 135960715 IC50 = 75 nM T48069 C36BQL 135960716 IC50 = 14 nM T48069 CVTF95 135960717 IC50 = 33 nM T48069 C01OML 135960718 IC50 = 27 nM T48069 C2G3JT 135960719 IC50 = 50 nM T48069 CI43OS 135960720 IC50 = 69 nM T48069 C6SZX2 135960721 IC50 = 37 nM T48069 C6E8WK 135960722 IC50 = 49 nM T48069 CZU46W 135960723 IC50 = 29 nM T48069 CUV5Q8 135960724 IC50 = 28 nM T48069 CFP18N 135960725 IC50 = 32 nM T48069 C4Z2CT 135960726 IC50 = 12 nM T48069 C3ST5C 135960727 IC50 = 40 nM T48069 CH4OX3 135960728 IC50 = 100 nM T48069 CVN7A3 135960729 IC50 = 82 nM T48069 CQ8BM7 135960730 IC50 = 100 nM T48069 CA26EL 135960731 IC50 = 37 nM T48069 C9GUD2 135960732 IC50 = 9 nM T48069 C3KU5W 135960733 IC50 = 16 nM T48069 CEGJ60 136007966 IC50 = 4000 nM T48069 CHA4N2 136013680 IC50 > 10 nM T48069 CLN6Y8 136026516 IC50 > 100000 nM T48069 CKC95O 136036546 IC50 = 38 nM T48069 C4FK8L 136036547 IC50 = 83 nM T48069 CB10LV 136036548 IC50 = 75 nM T48069 CB6M9H 136036549 IC50 = 172 nM T48069 C8SC9X 136036550 IC50 = 190 nM T48069 CA5QS9 136036551 IC50 = 480 nM T48069 C2HPZ1 136036552 IC50 = 1510 nM T48069 CN39EZ 136036553 IC50 = 360 nM T48069 CEL84G 136036554 IC50 = 82 nM T48069 CSW7U3 136036555 IC50 = 622 nM T48069 CSU7G4 136036556 IC50 = 360 nM T48069 CE2M1I 136036557 IC50 = 66 nM T48069 CELC04 136036558 IC50 = 243 nM T48069 C5JQY2 136036559 IC50 = 160 nM T48069 CYNE35 136036560 IC50 = 110 nM T48069 CU1HK5 136036561 IC50 = 680 nM T48069 CA6HK4 136036562 IC50 = 68 nM T48069 CY89TN 136036563 IC50 = 91 nM T48069 CE4D8Z 136036564 IC50 = 330 nM T48069 CT06IP 136036565 IC50 = 82 nM T48069 C0S7AP 136036566 IC50 = 96 nM T48069 CJ6Y9Q 136036567 IC50 = 796 nM T48069 CG89TM 136036568 IC50 = 290 nM T48069 C2VW7A 136036569 IC50 = 270 nM T48069 CQ9EY0 136036570 IC50 = 197 nM T48069 C74CYM 136036571 IC50 = 510 nM T48069 CL5F7Z 136036572 IC50 = 96 nM T48069 C7PS9L 136036573 IC50 = 630 nM T48069 CS8RA1 136066051 IC50 = 9 nM T48069 CN9WA6 136066052 IC50 = 319 nM T48069 CUE5X4 136086708 IC50 = 27 nM T48069 C80OJT 136086709 IC50 = 26 nM T48069 CY79BE 136086710 IC50 = 16 nM T48069 C2V8WH 136086711 IC50 = 38 nM T48069 C1EAF5 136086712 IC50 = 41 nM T48069 C5M6UO 136086713 IC50 = 30 nM T48069 CNEF50 136086718 IC50 = 17 nM T48069 CE9A5G 136086719 IC50 = 100 nM T48069 C27XOJ 136086720 IC50 = 28 nM T48069 C0K7PC 136086721 IC50 = 62 nM T48069 CC1DW7 136086722 IC50 = 210 nM T48069 C14APV 136086723 IC50 = 175 nM T48069 C3N5RQ 136086724 IC50 = 270 nM T48069 CJAY41 136117930 IC50 > 10000 nM T48069 CYJ53H 136117932 IC50 = 1790 nM T48069 CH68YK 136117933 IC50 = 3500 nM T48069 C7OB8V 136117934 IC50 = 440 nM T48069 CG0O9Q 136117981 IC50 = 4800 nM T48069 CC68KV 136117982 IC50 = 1700 nM T48069 CHE1L2 136117983 IC50 = 860 nM T48069 C31LFV 136117984 IC50 = 660 nM T48069 CP52YM 136117985 IC50 = 730 nM T48069 C6Y0OF 136117986 IC50 = 3300 nM T48069 C98UOE 136117987 IC50 = 5400 nM T48069 CS2N5H 136117988 IC50 = 570 nM T48069 C96OXH 136117989 IC50 = 13000 nM T48069 C31PNH 136117990 IC50 > 25000 nM T48069 CN0Q9H 136117991 IC50 = 3100 nM T48069 C69JHW 136117992 IC50 = 530 nM T48069 C5QEC7 136117993 IC50 > 25000 nM T48069 C4MSI6 136117994 IC50 = 1400 nM T48069 CH0SE6 136117995 IC50 > 25000 nM T48069 C0FY6E 136117996 IC50 > 25000 nM T48069 C92WUZ 136117997 IC50 = 590 nM T48069 CC74IA 136117998 IC50 > 25000 nM T48069 CWT49K 136117999 IC50 > 25000 nM T48069 CY96XL 136118000 IC50 = 1300 nM T48069 CNZY40 136118001 IC50 = 2200 nM T48069 C81WBZ 136118002 IC50 > 25000 nM T48069 CJ1DX7 136118003 IC50 = 530 nM T48069 C9SP6T 136118004 IC50 = 3500 nM T48069 C63VTD 136118015 IC50 = 1400 nM T48069 CL08HS 136118016 IC50 = 5100 nM T48069 CTSB03 136118017 IC50 = 3100 nM T48069 CS4TE6 136123410 IC50 = 830 nM T48069 C48DLS 136123445 IC50 = 68 nM T48069 C8D2FJ 136126667 IC50 = 30000 nM T48069 CSFU87 136164059 IC50 = 1300 nM T48069 C5FOH7 136164060 IC50 = 1550 nM T48069 CB9XQ1 136164061 IC50 = 5210 nM T48069 CIR40T 136164062 IC50 = 32 nM T48069 CD3F6B 136164063 IC50 = 32 nM T48069 C4YK0X 136164064 IC50 = 71 nM T48069 C19XOR 136164065 IC50 = 42 nM T48069 CD0G5X 136164066 IC50 = 330 nM T48069 C67AIH 136164067 IC50 = 410 nM T48069 CBU8W6 136164068 IC50 = 29 nM T48069 CG72LD 136164069 IC50 = 920 nM T48069 C7JX3S 136164070 IC50 = 2060 nM T48069 C1YUD0 136219394 IC50 > 10 nM T48069 CIU8W3 136254389 IC50 > 10 nM T48069 CE75QD 137321162 IC50 = 2100 nM T48069 C25ERN 137631967 IC50 > 1000 nM T48069 CI1E8V 137634241 IC50 = 6020 nM T48069 C06JRX 137637094 IC50 > 1000 nM T48069 C1DK0P 137651391 IC50 > 1000 nM T48069 C4HXK3 137655943 IC50 = 10 nM T48069 CV5H3Z 137657932 IC50 > 100 nM T48069 CUXO19 138617501 IC50 > 1000 nM T48069 CLRW84 139434103 EC50 = 840 nM T48069 CB6F5R 139434105 EC50 = 1800 nM T48069 C7FBY1 139434107 EC50 = 250 nM T48069 CJIH42 139434200 EC50 = 270 nM T48069 C4ID6F 139442949 EC50 = 220 nM T48069 CO9P7G 145351804 IC50 > 1000 nM T48069 C6VB3O 145925651 IC50 >= 5000 nM T48069 C4HB8M 145949394 IC50 = 4670 nM T48069 CB3Z1W 145949428 IC50 = 40 nM T48069 C5VSC7 145956704 IC50 = 6200 nM T48069 CRMN13 145963949 Ki = 2850 nM T48069 CI1UV7 145965620 Ki = 2610 nM T48069 C3YGN7 145966332 Ki = 2870 nM T48069 CHY74R 145966422 Ki = 2390 nM T48069 CZ38PG 145966502 IC50 > 1000000 nM T48069 C0G8ED 145966828 IC50 > 1000000 nM T48069 C4LHS5 145967074 Ki = 1920 nM T48069 COZA32 145967334 Ki = 540 nM T48069 CDNC31 145967951 IC50 > 500 nM T48069 C2J0VU 145968689 Ki = 3400 nM T48069 CW8UY6 145972402 Ki = 890 nM T48069 CKQ46V 145972976 Ki = 2100 nM T48069 CH5E2D 145973277 IC50 > 1000000 nM T48069 CTPQ06 145973553 Ki = 4560 nM T48069 CIKF18 145973791 Ki = 3560 nM T48069 CIWU86 145974353 Ki = 320 nM T48069 C5HB7J 145975494 IC50 > 1000000 nM T48069 CI7S4L 145976764 Ki = 4600 nM T48069 C69INU 145977311 Ki = 6180 nM T48069 C15XGN 145977927 Ki = 280 nM T48069 C46QAV 145977992 Ki = 3540 nM T48069 C6JBH1 145978562 Ki = 8930 nM T48069 C2MD1Q 155513187 IC50 > 10000 nM T48069 C3VTM7 155519139 IC50 = 6660 nM T48069 CM0U3I 155534552 IC50 = 109 nM T48069 CE46SL 155540854 IC50 = 10310 nM T48069 C5O4JM 155540856 IC50 = 3280 nM T48069 C0F5BN 155542940 IC50 = 434 nM T48069 CGVU70 155554426 IC50 > 30000 nM T48069 D00ATA 5908088 IC50 > 100000 nM T48069 D00ERW 44444843 Ki > 991 nM T48069 D00TBD 10461815 IC50 > 10000 nM T48069 D04ZWF 53396311 IC50 > 2000 nM T48069 D05RFO 24180536 IC50 = 90 nM T48069 D06HVH 54613583 IC50 > 10000 nM T48069 D06LJL 9916282 IC50 = 13000 nM T48069 D06NMZ 9825149 IC50 = 323 nM T48069 D06PJW 25182616 IC50 = 2 nM T48069 D06QWO 14824655 IC50 > 10 ug.mL-1 T48069 D07ADX 54764565 IC50 = 307 nM T48069 D07OSK 6419834 IC50 > 100000 nM T48069 D07SRX 9797919 IC50 > 10000 nM T48069 D08HFG 24809764 IC50 > 10000 nM T48069 D08HGK 3149447 IC50 > 100000 nM T48069 D09HVH 135566652 IC50 > 10 nM T48069 D09RYV 9911652 IC50 = 22000000 nM T48069 D09TNR 9850161 IC50 > 10000 nM T48069 D0A1CM 5281855 IC50 = 250 nM T48069 D0A4XJ 5289418 IC50 > 100000 nM T48069 D0B4SU 9549305 IC50 < 1000 nM T48069 D0C2GE 67161540 IC50 = 2700 nM T48069 D0E4LC 44581765 IC50 = 250 nM T48069 D0EE6A 6398883 IC50 > 10000 nM T48069 D0G3SZ 6918469 IC50 = 4.9 ug.mL-1 T48069 D0HE0E 5941540 IC50 > 100000 nM T48069 D0L7MM 43680262 IC50 = 4500 nM T48069 D0M4SY 135440466 IC50 = 100 nM T48069 D0NH7M 5328760 IC50 = 61 nM T48069 D0P6JS 11675054 IC50 > 10000 nM T48069 D0Q3EW 9549303 IC50 = 591 nM T48069 D0Q3KS 9957049 IC50 > 10000 nM T48069 D0R2WK 16038120 IC50 = 0.35 nM T48069 D0U3WQ 9817165 IC50 > 30000 nM T48069 D0W9KO 43743432 IC50 = 1500 nM T48069 D0Y0ES 3707 IC50 = 5300 nM T21307 D01BYB 5957 IC50 = 2800 nM T21307 D0E6XR 3062316 IC50 > 50000 nM T21307 D0EG1I 9926791 IC50 > 10000 nM T21307 D02NNV 3038525 IC50 > 5000 nM T21307 D03HUX 49792852 IC50 > 10000 nM T21307 D03LWG 53235510 IC50 > 10000 nM T21307 D07EHV 44814409 IC50 > 10000 nM T21307 D07HPJ 11476171 IC50 > 10000 nM T21307 D0E3TC 44259 IC50 = 150 nM T21307 D0O0LS 25141092 IC50 > 10000 nM T21307 D0O6WV 24794418 IC50 > 2000 nM T21307 D0P1CV 46191454 IC50 > 10000 nM T21307 D0Q9UX 16718576 IC50 > 10000 nM T21307 D03BNU 59604787 IC50 > 10000 nM T21307 D0LF0O 135441202 IC50 > 50000 nM T21307 D0R1JI 5281847 IC50 = 5400 nM T21307 D0T3ME 156422 IC50 > 30000 nM T21307 CK1GM9 7005 IC50 > 100000 nM T21307 CU5YR9 30386 IC50 = 85000 nM T21307 CK3F2W 145879 IC50 = 87000 nM T21307 CJ7NR2 176962 IC50 = 4500 nM T21307 CJGW48 202978 IC50 > 40000 nM T21307 C1EB0M 461195 IC50 = 1090 nM T21307 CC31FE 512549 IC50 = 180 nM T21307 C2ZN0H 512561 IC50 = 300 nM T21307 C0YIB2 512562 IC50 = 40 nM T21307 CEM7X3 612268 IC50 > 200000 nM T21307 CVN83J 656950 IC50 > 10000 nM T21307 C03XPN 1494312 IC50 = 6000 nM T21307 C1SVD2 2132479 IC50 = 9800 nM T21307 C5EW4Z 3264448 IC50 = 5200 nM T21307 CJWX69 3848929 IC50 = 2500 nM T21307 C7I9GF 4274924 IC50 > 200000 nM T21307 CL5I2U 5330279 IC50 > 10000 nM T21307 CG17TN 6914611 IC50 > 50000 nM T21307 C7E2QK 6914613 IC50 > 10000 nM T21307 CA3BD9 9821424 IC50 = 130 nM T21307 C7YVW1 9826115 EC50 = 28 nM T21307 CRC65X 9863786 IC50 > 30000 nM T21307 CM5Z8X 9869943 IC50 > 1000 nM T21307 C12PKF 9871380 IC50 > 25000 nM T21307 C18HKQ 9885748 IC50 > 100000 nM T21307 C2Y3WG 9907612 IC50 = 1300 nM T21307 CS5KX9 9938299 IC50 > 10000 nM T21307 CJO47T 9948405 IC50 > 10000 nM T21307 CO5L1Q 9971229 IC50 > 200000 nM T21307 CV28XH 9979332 IC50 = 600 nM T21307 CV8I5X 9999342 IC50 > 10000 nM T21307 CPSY37 10001536 IC50 = 8100 nM T21307 C7Z1FR 10007353 IC50 = 8 nM T21307 C7YD1X 10048045 IC50 > 25000 nM T21307 CT70MI 10049465 IC50 = 1600 nM T21307 C93UVK 10092544 IC50 = 400 nM T21307 CAT54X 10106198 IC50 = 70000 nM T21307 C0R5AX 10215912 IC50 > 50000 nM T21307 C5TQ7X 10247543 IC50 > 10000 nM T21307 CB2GC4 10250350 IC50 = 3100 nM T21307 CP38GX 10313607 IC50 = 49 nM T21307 CQK48V 10339752 IC50 = 360 nM T21307 C7HBP6 10429593 IC50 > 10000 nM T21307 C62KGB 10430385 IC50 = 400 nM T21307 CTJ8K5 10430386 IC50 = 700 nM T21307 C69ZOB 10453611 IC50 = 8 nM T21307 CB86LA 10456600 IC50 = 9200 nM T21307 C3P7QD 10467496 IC50 > 200000 nM T21307 C2WQ8M 10473563 IC50 > 10000 nM T21307 CK63DE 10621161 IC50 = 90000 nM T21307 C2W5RC 11235063 IC50 > 50000 nM T21307 C6C3JX 11281930 IC50 > 10000 nM T21307 CN4ED9 11292790 IC50 = 20000 nM T21307 CBOP58 11293798 Ki = 880 nM T21307 CRTG16 11359538 IC50 = 17000 nM T21307 CDAR63 11361892 IC50 = 9600 nM T21307 C26BZX 11362471 Ki = 1570 nM T21307 CWXB93 11397177 Ki > 10000 nM T21307 C0APW4 11422034 IC50 > 10000 nM T21307 CJC95A 11454205 IC50 > 10000 nM T21307 CS4MT5 11495655 IC50 = 2600 nM T21307 CT9V3D 11496376 IC50 > 400000 nM T21307 C59BEW 11517184 IC50 = 700 nM T21307 CEV61O 11525487 IC50 = 1500 nM T21307 C7HMO6 11526786 IC50 > 200000 nM T21307 CTG83F 11539329 Ki > 8400 nM T21307 C78BJQ 11554437 IC50 = 1400 nM T21307 CACS26 11561968 Ki > 2000 nM T21307 C87TNU 11575548 Ki = 96 nM T21307 CO9KP5 11583459 IC50 > 10000 nM T21307 CMIL86 11590363 Ki > 8400 nM T21307 CA07WQ 11604613 IC50 = 700 nM T21307 C5ER7L 11632412 IC50 = 90000 nM T21307 CK34LS 11632737 IC50 > 50000 nM T21307 C6UT5Q 11632886 IC50 = 1400 nM T21307 C9T6SC 11640926 Ki > 8400 nM T21307 C4GTZ8 11645322 IC50 > 20000 nM T21307 CL7NV5 11654763 IC50 = 8000 nM T21307 CJ9KN7 11683817 IC50 > 10000 nM T21307 CU0E8O 11690457 Ki > 2000 nM T21307 CC03XG 11718461 IC50 = 800 nM T21307 CZ3Q7B 11719115 IC50 = 9000 nM T21307 C9JT4S 11847343 IC50 > 10000 nM T21307 C8E4TS 11992146 IC50 = 126 nM T21307 C90WYL 12773710 IC50 = 26000 nM T21307 C3YRU7 15295578 IC50 = 8900 nM T21307 CLN43D 15366651 IC50 = 22500 nM T21307 CA1PQ3 15604675 IC50 = 1700 nM T21307 C34YWT 15604761 IC50 = 1100 nM T21307 C0B7EG 15604763 IC50 = 2300 nM T21307 CO0Z5E 15604765 IC50 = 1400 nM T21307 CYR2G7 15604766 IC50 = 160 nM T21307 CL9J8B 15604844 IC50 = 320 nM T21307 CJ0RV5 15951573 IC50 = 760 nM T21307 C4JN6B 15951575 IC50 = 1700 nM T21307 CO3QF7 15951576 IC50 = 520 nM T21307 C1ASL6 15951577 IC50 = 1300 nM T21307 CU6J8N 15951675 IC50 = 770 nM T21307 C1LDI3 15951676 IC50 = 820 nM T21307 CLEV74 15951677 IC50 = 1700 nM T21307 CF70GK 15951678 IC50 = 7400 nM T21307 CPQA87 15951768 IC50 = 620 nM T21307 C37CMO 15951769 IC50 = 2700 nM T21307 CS5NH9 15951859 IC50 > 10000 nM T21307 CL5Y4G 15951863 IC50 = 2700 nM T21307 CVJ6R3 15951865 IC50 = 3000 nM T21307 CB0AW7 15951956 IC50 = 7000 nM T21307 C1T7CM 15951958 IC50 = 1500 nM T21307 C8R0NU 15952051 IC50 = 440 nM T21307 CL1H4E 15952054 IC50 = 3400 nM T21307 COV71G 15952058 IC50 > 20000 nM T21307 CHS9Z0 15952150 IC50 = 9700 nM T21307 CQW20R 15952154 IC50 > 20000 nM T21307 C2WS0K 15952155 IC50 = 1500 nM T21307 COU61A 15952243 IC50 > 20000 nM T21307 CR9S6I 15952246 IC50 > 20000 nM T21307 CEAH07 15952340 IC50 > 10000 nM T21307 CX2IV4 15952341 IC50 > 20000 nM T21307 C1M4EL 15952435 IC50 = 750 nM T21307 C8PZ7K 15952436 IC50 = 770 nM T21307 CY0G9I 15952825 IC50 = 2900 nM T21307 C3BA8V 15952827 IC50 = 12000 nM T21307 C2LQJ6 15952933 IC50 = 3000 nM T21307 CV6OQ1 15952934 IC50 = 7700 nM T21307 C9TU1O 16046126 IC50 > 1000 nM T21307 CZHJ34 16058637 IC50 > 50000 nM T21307 CKV4G1 16079040 IC50 = 6700 nM T21307 CKX2L7 16085320 IC50 > 400000 nM T21307 CVZK29 16223008 IC50 > 50000 nM T21307 CUR7H3 16719862 IC50 = 66 nM T21307 C1OH3G 16719968 IC50 = 56 nM T21307 C1JHO9 16719970 IC50 = 48 nM T21307 CX7E5U 16719971 IC50 = 83 nM T21307 C6XYB4 16719973 IC50 = 76 nM T21307 CVC65T 16719974 IC50 = 52 nM T21307 C7V0YT 16719976 IC50 = 30 nM T21307 CCO4R6 16720087 IC50 = 25 nM T21307 C5MPI6 16720090 IC50 = 606 nM T21307 CJ2CW0 16720091 IC50 = 37 nM T21307 CP9HE8 16720093 IC50 = 32 nM T21307 CLW0F1 16720095 IC50 = 30 nM T21307 C8GOE5 16720200 IC50 = 50 nM T21307 CY7IM4 16720202 IC50 = 171 nM T21307 CT4LF5 16720203 IC50 = 62 nM T21307 C81FSH 16720205 IC50 = 51 nM T21307 CGO45Z 16720207 IC50 = 55 nM T21307 C8DKE0 16720208 IC50 = 41 nM T21307 C8BJ4X 16720315 IC50 = 22 nM T21307 C9PH0U 16720316 IC50 = 15 nM T21307 C2BKD4 16720318 IC50 = 17 nM T21307 CR2PQ1 16720319 IC50 = 46 nM T21307 CSON67 16720432 IC50 = 608 nM T21307 C8DI3J 16720542 IC50 = 56 nM T21307 CVS0T5 17754396 IC50 > 10000 nM T21307 C8AH1I 17758019 IC50 = 35800 nM T21307 C1GKL6 17758020 IC50 > 40000 nM T21307 CIE58R 17758239 IC50 = 62700 nM T21307 CO6LR5 17758240 IC50 > 40000 nM T21307 CWH37T 17758574 IC50 = 87100 nM T21307 C57NRL 17759787 IC50 = 40100 nM T21307 CX4N3K 17881612 IC50 = 42000 nM T21307 CNDF83 20066922 IC50 = 4500 nM T21307 CR64BI 20805054 IC50 = 3800 nM T21307 CH4B5K 21081523 IC50 > 5000 nM T21307 C25UKC 21081761 IC50 > 10000 nM T21307 CS31DN 21399939 IC50 > 200000 nM T21307 CHKM46 21590533 IC50 = 90000 nM T21307 CNKF46 21590534 IC50 = 90000 nM T21307 CW6OB1 23627212 IC50 > 9000 nM T21307 CG6D4M 23647319 IC50 > 10000 nM T21307 CY8Z7X 23647330 IC50 > 10000 nM T21307 C4XD8H 23647348 IC50 > 10000 nM T21307 CDMI50 23661564 IC50 = 290 nM T21307 C13XMS 23661565 IC50 = 10100 nM T21307 C6ZTS8 23661566 IC50 = 10 nM T21307 CV9U8E 24745781 IC50 > 10000 nM T21307 C7YG1N 24759534 IC50 = 55000 nM T21307 C2UOE0 24766030 IC50 > 50000 nM T21307 CJUK39 24770517 IC50 > 10000 nM T21307 C9PA0M 24807809 IC50 > 200000 nM T21307 CCP2M3 24822704 IC50 > 50000 nM T21307 CM28WD 24825721 IC50 > 10000 nM T21307 CC9V2Y 24882562 IC50 = 2 nM T21307 C13QYB 24884503 IC50 > 2000 nM T21307 CY8L7E 24896769 IC50 > 10000 nM T21307 C4EG8R 24993189 IC50 > 10000 nM T21307 CVQS96 25052767 IC50 = 4.3 nM T21307 CAO8Q2 25064527 IC50 = 72 nM T21307 C0GX6V 25064951 IC50 = 27 nM T21307 CBZS28 25065155 IC50 = 900 nM T21307 C0JT3O 25065992 IC50 = 32 nM T21307 CB5TY4 25066206 IC50 = 5 nM T21307 CX2J3S 25066411 IC50 = 16 nM T21307 CM04RX 25066412 IC50 = 2500 nM T21307 CG34VQ 25066413 IC50 = 80 nM T21307 CJRG97 25066414 IC50 = 96 nM T21307 CN9SJ7 25066415 IC50 = 5 nM T21307 C7IM8Q 25066416 IC50 = 12 nM T21307 C57TQU 25066617 IC50 = 15 nM T21307 C7BI0O 25066619 IC50 = 160 nM T21307 CD8B9A 25118220 IC50 = 5.7 nM T21307 CY14DU 25119291 IC50 = 7 nM T21307 C4DA6F 25205591 IC50 = 8200 nM T21307 C4VD0S 25205757 IC50 = 88000 nM T21307 CLFM35 25206064 IC50 = 4500 nM T21307 CXR81L 25206065 IC50 > 100000 nM T21307 C1RV7S 25206391 IC50 = 5000 nM T21307 C8T6PZ 25207350 IC50 > 100000 nM T21307 CSGI69 25207352 IC50 > 100000 nM T21307 C8A6HJ 25207353 IC50 > 100000 nM T21307 CPL2A7 25207355 IC50 = 65000 nM T21307 C23OYR 25207516 IC50 > 100000 nM T21307 CCV57R 25207519 IC50 = 2300 nM T21307 CNG96H 25210579 IC50 > 10000 nM T21307 CRO09K 25211064 IC50 > 100000 nM T21307 C4T7YX 25218756 IC50 > 50000 nM T21307 CWS37O 42618140 IC50 > 25118.86 nM T21307 C2JV3O 42618143 IC50 > 25118.86 nM T21307 CG01BO 42618144 IC50 > 25118.86 nM T21307 CXI08R 42646194 IC50 = 150 nM T21307 C42DXS 42646445 IC50 = 12 nM T21307 C9E2UW 42646446 IC50 = 50 nM T21307 CAFO97 42646698 IC50 < 3 nM T21307 CFEW87 42646706 IC50 < 3 nM T21307 C48USC 44143344 IC50 > 400000 nM T21307 C8YN5P 44143370 IC50 = 63000 nM T21307 C9CWO1 44143371 IC50 > 200000 nM T21307 C26XFL 44143372 IC50 > 200000 nM T21307 C5SEQ2 44143373 IC50 = 131000 nM T21307 C1X5NY 44143506 IC50 > 40000 nM T21307 CIX56K 44143507 IC50 > 40000 nM T21307 C18SJA 44143508 IC50 > 40000 nM T21307 CV7A5Y 44143509 IC50 = 15000 nM T21307 C20XQB 44143510 IC50 > 40000 nM T21307 CZ7QP2 44143511 IC50 > 40000 nM T21307 CV87MH 44143512 IC50 > 40000 nM T21307 CL4EA1 44143513 IC50 = 5400 nM T21307 C54WOA 44143514 IC50 > 20000 nM T21307 CK8Y0X 44143515 IC50 > 20000 nM T21307 C1YS4B 44143516 IC50 > 20000 nM T21307 CG93PA 44143517 IC50 > 20000 nM T21307 CJ03IG 44143518 IC50 > 20000 nM T21307 CX76PQ 44143519 IC50 = 1500 nM T21307 C8Z7ID 44143520 IC50 = 3000 nM T21307 CH87PN 44143521 IC50 = 1700 nM T21307 CX2V9R 44143522 IC50 = 4400 nM T21307 CKG43S 44143523 IC50 = 930 nM T21307 CG29TE 44143524 IC50 = 1800 nM T21307 CK47XB 44143525 IC50 = 760 nM T21307 CJAK48 44143526 IC50 = 620 nM T21307 CM86PK 44143527 IC50 = 83 nM T21307 CK6EJ9 44143528 IC50 = 120 nM T21307 CW3M7Y 44143529 IC50 = 72 nM T21307 C4ES7R 44143530 IC50 = 333 nM T21307 CC9SL5 44143531 IC50 = 34 nM T21307 C94BQU 44143532 IC50 = 17 nM T21307 CGY5K0 44143533 IC50 = 35 nM T21307 CFP1N7 44143534 IC50 = 124 nM T21307 CQFJ89 44143535 IC50 = 21 nM T21307 CI0JH3 44143536 IC50 = 31 nM T21307 C1MFQ2 44143537 IC50 = 45 nM T21307 C6E4SD 44143538 IC50 = 44 nM T21307 CT5YO0 44143539 IC50 = 250 nM T21307 C50UIG 44143540 IC50 = 1300 nM T21307 C87FZR 44143541 IC50 = 480 nM T21307 CVQO95 44143542 IC50 = 2600 nM T21307 CO9L3N 44143543 IC50 = 260 nM T21307 C32INU 44143544 IC50 = 1200 nM T21307 C3WJM7 44143545 IC50 = 140 nM T21307 C65WQK 44143546 IC50 = 1000 nM T21307 CI9AW3 44143547 IC50 = 210 nM T21307 C3U0QC 44143548 IC50 > 10000 nM T21307 C40JYN 44143549 IC50 = 1200 nM T21307 C3W8QK 44143550 IC50 = 550 nM T21307 CNVY08 44143551 IC50 = 4000 nM T21307 CVH21S 44143552 IC50 = 580 nM T21307 C9PMI2 44143553 IC50 = 3000 nM T21307 CEXA13 44143554 IC50 = 4000 nM T21307 C5Z1RX 44143555 IC50 > 10000 nM T21307 C9FXA4 44143556 IC50 > 10000 nM T21307 CH7EM3 44143557 IC50 = 6900 nM T21307 CNA95E 44143558 IC50 = 270 nM T21307 CH2F9K 44143559 IC50 = 190 nM T21307 C04QTA 44143560 IC50 = 29 nM T21307 CIH05K 44143561 IC50 = 320 nM T21307 C7QM5O 44143562 IC50 = 35 nM T21307 CUK52C 44143563 IC50 = 52 nM T21307 C7LV5P 44143564 IC50 = 530 nM T21307 CA52CH 44143565 IC50 = 690 nM T21307 CW7Y8Z 44143566 IC50 = 560 nM T21307 C3HC8V 44143567 IC50 = 310 nM T21307 CC4QR6 44143568 IC50 = 1200 nM T21307 CLW80F 44160269 IC50 = 22000 nM T21307 CK73NR 44219749 IC50 > 50000 nM T21307 CCZ20U 44224182 IC50 = 45 nM T21307 CI58SN 44224183 IC50 = 20 nM T21307 C4QM3P 44224184 IC50 = 15 nM T21307 C52INR 44269421 IC50 > 200000 nM T21307 CZ4VX0 44405504 IC50 > 400000 nM T21307 CGI5L7 44405938 IC50 > 20000 nM T21307 C0G3WF 44405939 IC50 > 20000 nM T21307 CR3Q7Z 44405940 IC50 > 20000 nM T21307 C79WRL 44405941 IC50 > 20000 nM T21307 C0XZ8K 44406013 IC50 > 20000 nM T21307 CS3K1P 44406014 IC50 = 16000 nM T21307 CC93JP 44406018 IC50 > 20000 nM T21307 CCRZ12 44406074 IC50 > 20000 nM T21307 C9CO8R 44440882 IC50 = 2700 nM T21307 CCG3T8 44440883 IC50 > 40000 nM T21307 C7NJ9V 44440884 IC50 > 40000 nM T21307 CQ3IL2 44440885 IC50 = 1100 nM T21307 CC9FV1 44440886 IC50 > 40000 nM T21307 C6ULE3 44440887 IC50 > 40000 nM T21307 CPID20 44441112 IC50 > 200000 nM T21307 C32SJG 44441113 IC50 > 200000 nM T21307 C4WON2 44441114 IC50 = 53000 nM T21307 CE6W0H 44441115 IC50 > 200000 nM T21307 C4YN9A 44441116 IC50 = 6600 nM T21307 CDG95H 44441117 IC50 = 170000 nM T21307 CV37CM 44441118 IC50 = 19000 nM T21307 CL2B4M 44441119 IC50 = 28000 nM T21307 C7ESN6 44441120 IC50 = 12000 nM T21307 CNIE57 44441121 IC50 = 1100 nM T21307 C53DPU 44441122 IC50 > 200000 nM T21307 C8VZ3X 44441123 IC50 > 200000 nM T21307 CV34IO 44441124 IC50 = 1000 nM T21307 C8UNW4 44441126 IC50 = 5800 nM T21307 CB34LX 44441127 IC50 = 170000 nM T21307 CHMZ24 44441128 IC50 = 130000 nM T21307 C48QPX 44441129 IC50 = 47000 nM T21307 CPHD54 44441130 IC50 > 200000 nM T21307 CYK97G 44441131 IC50 > 200000 nM T21307 C2QJX7 44441132 IC50 > 200000 nM T21307 CJ19HU 44441133 IC50 = 88000 nM T21307 CCS6M4 44441134 IC50 = 130000 nM T21307 CQ4F6R 44441135 IC50 > 200000 nM T21307 C9BCE4 44441136 IC50 = 2200 nM T21307 C7DT4K 44441137 IC50 = 2200 nM T21307 CMJ84G 44441139 IC50 = 16000 nM T21307 C8C3GD 44441140 IC50 = 7100 nM T21307 CVM3H5 44441141 IC50 = 64000 nM T21307 C13EIV 44441142 IC50 > 200000 nM T21307 CO7I2H 44441143 IC50 = 3000 nM T21307 CT9CU2 44441144 IC50 = 5900 nM T21307 CNB18G 44441146 IC50 > 200000 nM T21307 C9URB7 44441149 IC50 = 5100 nM T21307 CU9I3O 44441151 IC50 = 29300 nM T21307 CMQ2D8 44441152 IC50 = 7090 nM T21307 C7G0FT 44441155 IC50 = 3270 nM T21307 CPB8Y7 44441158 IC50 = 13000 nM T21307 CSA12W 44450544 IC50 = 110000000 nM T21307 CUMN81 44454600 IC50 = 5 nM T21307 CW8C2F 44454601 IC50 = 3 nM T21307 CI3RB0 44454629 IC50 = 2 nM T21307 C63NKR 44454631 IC50 = 2 nM T21307 CG3R9U 44454652 IC50 = 5 nM T21307 CEK6I3 44454653 IC50 = 9 nM T21307 CKVT48 44454654 IC50 = 19 nM T21307 CB9WQ2 44454679 IC50 = 4 nM T21307 C27FGN 44454680 IC50 = 3 nM T21307 CBFO39 44454683 IC50 = 7 nM T21307 CA1Q6N 44454704 IC50 = 45 nM T21307 CM2XI4 44454705 IC50 = 46 nM T21307 CB7Y0X 44454706 IC50 = 12 nM T21307 CG0PJ9 44454732 IC50 = 5 nM T21307 C75NDI 44454733 IC50 = 20 nM T21307 C48HGY 44517741 IC50 = 1 nM T21307 CA7TD4 44517742 IC50 = 16 nM T21307 C4WRN5 44541014 IC50 = 6.5 nM T21307 C3NZV6 44543658 IC50 = 1300 nM T21307 CJY8S0 44570884 IC50 > 5000 nM T21307 C1STH4 44574421 IC50 = 2400 nM T21307 CZR3L0 44574422 IC50 = 670 nM T21307 CU8G1L 44574423 IC50 = 1600 nM T21307 CAGP18 44574424 IC50 = 2300 nM T21307 CDZC64 44574425 IC50 = 3800 nM T21307 CEUK81 44574469 IC50 = 1300 nM T21307 CA28XU 44574873 IC50 > 100000 nM T21307 C2VY0T 44574928 IC50 = 81000 nM T21307 CR2YO5 44574929 IC50 = 9300 nM T21307 C5KHD2 44574930 IC50 = 33000 nM T21307 CV31ER 44574931 IC50 = 49000 nM T21307 CFHW18 44574932 IC50 = 14000 nM T21307 CWV59R 44574933 IC50 = 380 nM T21307 C8GTE4 44574982 IC50 = 5500 nM T21307 C1TAL5 44574983 IC50 = 24000 nM T21307 CQS7H5 44575024 IC50 = 5300 nM T21307 CU38NY 44575025 IC50 > 100000 nM T21307 C2E3LA 44575072 IC50 = 2600 nM T21307 CCL85F 44575073 IC50 = 5800 nM T21307 CF6Y2A 44575074 IC50 = 6600 nM T21307 CV54BF 44575124 IC50 = 3700 nM T21307 CHT5M7 44575125 IC50 = 3600 nM T21307 CJX06P 44575126 IC50 = 5300 nM T21307 CE8FC7 44575127 IC50 = 5400 nM T21307 CG7BV1 44575128 IC50 = 9100 nM T21307 C5Z3LI 44591740 IC50 = 13000 nM T21307 COY57J 44592504 IC50 = 2500 nM T21307 CV8F0R 44593854 IC50 = 61 nM T21307 C28QLM 44605035 IC50 > 50000 nM T21307 C75XHS 44605037 IC50 > 50000 nM T21307 C8ZCP1 44631900 IC50 = 30 nM T21307 CU3RF1 45139989 IC50 > 10000 nM T21307 CQGZ06 45139991 IC50 > 10000 nM T21307 CY83PR 45267327 IC50 > 1000 nM T21307 C2I3QV 45267582 IC50 = 2 nM T21307 C7H0EZ 45267583 IC50 = 5 nM T21307 C9V6NQ 45267633 IC50 = 3500 nM T21307 CNA6Z4 45267641 IC50 = 3440 nM T21307 C75WAC 45268471 IC50 = 1040 nM T21307 CL3ZD2 45268500 IC50 = 14 nM T21307 C43MRK 45268501 IC50 = 450 nM T21307 C8WJ4I 45268513 IC50 = 1320 nM T21307 C84QFJ 45269074 IC50 > 1000 nM T21307 CN4TD8 45269319 IC50 = 6800 nM T21307 C0L3KN 45269326 IC50 = 41 nM T21307 CH59DU 45269365 IC50 = 1910 nM T21307 CVJ70Z 45269366 IC50 = 4600 nM T21307 C9NCR0 45269376 IC50 = 3100 nM T21307 C6B9VH 45270159 IC50 = 23 nM T21307 C59YDL 45271022 IC50 = 570 nM T21307 C9HO2X 45271028 IC50 > 20000 nM T21307 CG83KW 45271845 IC50 = 9 nM T21307 C92ZKY 45271846 IC50 = 14 nM T21307 C4C0TD 45271854 IC50 = 930 nM T21307 C6U1LK 45271859 IC50 = 5 nM T21307 C7D5FQ 45271878 IC50 = 1520 nM T21307 C04AVC 45271879 IC50 = 500 nM T21307 C0KFU4 45271889 IC50 = 570 nM T21307 CGOR36 45271890 IC50 > 20000 nM T21307 CK3F4V 45272705 IC50 = 28 nM T21307 CT7RV8 45272713 IC50 = 30 nM T21307 C3DH8I 45273358 IC50 = 540 nM T21307 C06JQE 45273683 IC50 = 2600 nM T21307 CC95PQ 45375865 IC50 > 50000 nM T21307 CEOQ27 45375866 IC50 > 50000 nM T21307 C5S8MA 45485083 IC50 > 8000 nM T21307 C79MHP 45485213 IC50 = 570 nM T21307 CW42YX 45487634 IC50 > 5000 nM T21307 C96BNW 46179972 IC50 > 50000 nM T21307 CKVS86 46224666 IC50 = 720 nM T21307 C27ALO 46224671 IC50 = 1400 nM T21307 C4WA0K 46224674 IC50 = 1600 nM T21307 CDR9W1 46224675 IC50 = 1900 nM T21307 CYZ63F 46224679 IC50 = 820 nM T21307 C2W4JR 46224682 IC50 = 310 nM T21307 CY3HW5 46224684 IC50 = 19 nM T21307 CI1J7P 46224686 IC50 = 9100 nM T21307 CEB98V 46224689 IC50 = 24000 nM T21307 CQW1M5 46224690 IC50 = 3400 nM T21307 C7KP1I 46224694 IC50 = 14000 nM T21307 C2UDM7 46224695 IC50 = 160 nM T21307 CEM0H4 46224696 IC50 = 56 nM T21307 CA74TK 46224697 IC50 = 35 nM T21307 CF9X8K 46224698 IC50 = 960 nM T21307 C9WY1E 46224700 IC50 = 5400 nM T21307 C56UCM 46224701 IC50 = 260 nM T21307 CX9I3N 46224703 IC50 = 49000 nM T21307 C6JD8T 46224704 IC50 = 37 nM T21307 C37YWV 46226031 IC50 > 50000 nM T21307 CB65AX 46226037 IC50 = 1900 nM T21307 C7XF6H 46226038 IC50 = 490 nM T21307 CEVW09 46226047 IC50 = 20 nM T21307 C01ASJ 46226048 IC50 = 41 nM T21307 CW41OF 46231423 IC50 = 22600 nM T21307 CML4R3 46231473 IC50 = 2000 nM T21307 CP7J3Z 46231474 IC50 = 31200 nM T21307 CJ72YD 46231475 IC50 = 15400 nM T21307 CGY19B 46231476 IC50 = 6000 nM T21307 CYM97E 46231477 IC50 = 84 nM T21307 C24VNP 46231531 IC50 = 1100 nM T21307 C0W2TG 46231532 IC50 = 350 nM T21307 C0E6YX 46231533 IC50 = 180 nM T21307 C2BF5K 46231534 IC50 = 180 nM T21307 CZ7PR4 46231583 IC50 = 180 nM T21307 CC5ET2 46231584 IC50 = 82 nM T21307 C4H5YX 46231585 IC50 = 290 nM T21307 CIBS16 46231638 IC50 = 220 nM T21307 C7ON5A 46233287 IC50 > 10000 nM T21307 COTJ39 46863083 IC50 = 60 nM T21307 C0F9RH 46863195 IC50 = 910 nM T21307 CD0YE5 46863197 IC50 = 10000 nM T21307 C5FMC8 46863199 IC50 = 4150 nM T21307 CLD1W7 46863317 IC50 = 4090 nM T21307 C64LIW 46863435 IC50 = 400 nM T21307 C0CXG9 46863436 IC50 = 820 nM T21307 CA4QB7 46863552 IC50 = 910 nM T21307 CO3P0J 46866604 IC50 < 50000 nM T21307 CLS29B 46872626 IC50 > 10000 nM T21307 CJOM49 46880136 IC50 = 17100 nM T21307 C0FD1O 46927902 IC50 = 400 nM T21307 C2B5XF 49765254 IC50 > 10000 nM T21307 C9L3XR 49838879 IC50 > 30000 nM T21307 CJZ5A0 49840306 IC50 > 10000 nM T21307 CF91RS 49843531 IC50 > 10000 nM T21307 CK4S8Y 49862001 IC50 = 27000 nM T21307 C1T4EX 49862002 IC50 = 15000 nM T21307 CY1V9B 49862003 IC50 = 33000 nM T21307 C4Q3DP 49862004 IC50 = 25000 nM T21307 CG6AV2 49862005 IC50 = 27000 nM T21307 C5F0MJ 49862049 IC50 = 35000 nM T21307 CT3P6K 49862050 IC50 = 43000 nM T21307 C9Q2PW 49862051 IC50 = 121000 nM T21307 C1P5ZG 49862052 IC50 = 26000 nM T21307 C10UDH 49862087 IC50 > 200000 nM T21307 C4LTF6 49862088 IC50 > 200000 nM T21307 CP3R9I 49862123 IC50 > 200000 nM T21307 CF5AB7 49862124 IC50 = 14000 nM T21307 C6BIP2 49862167 IC50 = 1800 nM T21307 C8R2CJ 49862702 IC50 > 200000 nM T21307 CDAX89 49862703 IC50 = 22000 nM T21307 CXE2I8 49862704 IC50 = 41000 nM T21307 COI1U3 49862778 IC50 = 120000 nM T21307 CHS56Y 49862779 IC50 = 12000 nM T21307 C62NDA 49862780 IC50 = 23000 nM T21307 C0GQX7 49862781 IC50 = 24000 nM T21307 C0SE7A 49862782 IC50 = 29000 nM T21307 CNT8C4 49867482 IC50 = 130 nM T21307 C2Y6QS 50938552 IC50 > 10000 nM T21307 C9NYP4 51036677 IC50 > 10000 nM T21307 C4WRY3 51037112 IC50 > 10000 nM T21307 CRI28Z 51037948 IC50 > 10000 nM T21307 C0QCK6 53235497 EC50 = 138 nM T21307 C4H2EJ 53235515 EC50 = 2.1 nM T21307 CCZX09 53246589 EC50 = 5.9 nM T21307 C0X2DB 53246706 EC50 = 29 nM T21307 C3CK1G 53246707 EC50 = 8.3 nM T21307 C1UPV2 53246708 EC50 = 9.8 nM T21307 C5BHK4 53246828 EC50 = 112 nM T21307 C6YWL8 53246831 EC50 = 6.9 nM T21307 CND1R5 53246955 EC50 = 15 nM T21307 CADY61 53251162 IC50 = 64 nM T21307 CCL72O 53251319 IC50 = 52 nM T21307 C6OTY5 53251320 IC50 = 22 nM T21307 CM03DF 53251321 IC50 = 110 nM T21307 CBV6I0 53251322 IC50 = 5.7 nM T21307 CJW3Q2 53251323 IC50 = 79 nM T21307 CLBC48 53251479 IC50 = 107 nM T21307 CR3ZM1 53251480 IC50 = 110 nM T21307 CN3FX4 53251481 IC50 = 39 nM T21307 CC2PN0 53251635 IC50 = 96 nM T21307 C8SC2X 53251787 IC50 = 21 nM T21307 CO3DV1 53251940 IC50 = 14 nM T21307 CZ92KP 53326866 EC50 = 4 nM T21307 C8ZRE3 53356518 IC50 = 13330 nM T21307 C8NA4L 53384644 IC50 > 30000 nM T21307 C6DA7C 53389527 EC50 = 7.4 nM T21307 CQ2P5I 53467419 IC50 = 400 nM T21307 CITN21 53475321 IC50 = 110 nM T21307 CT9AR0 54580390 IC50 = 2000 nM T21307 C5HQW3 54580391 IC50 = 2700 nM T21307 CA2ES1 54580392 IC50 = 3700 nM T21307 CK74QR 54580393 IC50 = 10700 nM T21307 CGQ1K6 54580426 IC50 = 2600 nM T21307 CV4EU2 54580427 IC50 = 40000 nM T21307 CYO5U8 54580428 IC50 = 210 nM T21307 CX1GH3 54580429 IC50 = 3800 nM T21307 C1RJB7 54580430 IC50 = 15000 nM T21307 C9I4AS 54580533 EC50 = 129 nM T21307 CZY4I9 54580537 EC50 = 234 nM T21307 C8E6RF 54580895 EC50 = 4.5 nM T21307 CB0IS4 54580896 EC50 = 1.1 nM T21307 C0NQ3B 54580897 EC50 = 11 nM T21307 C74CBA 54581389 IC50 = 20000 nM T21307 CK9CG3 54581390 IC50 = 12000 nM T21307 CJ65AU 54581391 IC50 = 36000 nM T21307 CEK63R 54581392 IC50 = 22000 nM T21307 CG9R6S 54581393 IC50 = 2600 nM T21307 C9S5IT 54581394 IC50 = 9900 nM T21307 C98BZJ 54581395 IC50 > 40000 nM T21307 CF8O9E 54581396 IC50 = 5200 nM T21307 CC7L4U 54581434 IC50 = 730 nM T21307 CC8KT1 54581435 IC50 = 2900 nM T21307 CT7HZ0 54581436 IC50 = 14000 nM T21307 C9ZKU6 54581952 EC50 = 724 nM T21307 C8WR1L 54581953 EC50 = 5.1 nM T21307 CX8HS6 54581954 EC50 = 3.6 nM T21307 CTD60M 54582407 IC50 = 50000 nM T21307 CH0D1V 54582408 IC50 > 50000 nM T21307 C6T3BJ 54582440 IC50 = 1500 nM T21307 CN5B9D 54582441 IC50 = 3600 nM T21307 C3V0BS 54582442 IC50 = 2500 nM T21307 CS7J4D 54582443 IC50 = 310 nM T21307 CPS08Z 54582444 IC50 = 700 nM T21307 CIFR35 54582445 IC50 = 103 nM T21307 CCYM61 54582533 EC50 = 6.5 nM T21307 C4AT5X 54582534 EC50 = 151 nM T21307 C8F9JB 54582875 EC50 = 13 nM T21307 CM7I5U 54582876 EC50 = 6.9 nM T21307 CV4A3T 54582877 EC50 = 28 nM T21307 CI6C1U 54583388 IC50 > 50000 nM T21307 CF2VO6 54583389 IC50 = 4000 nM T21307 CK4WD9 54583390 IC50 = 1500 nM T21307 C0NRW8 54583391 IC50 = 470 nM T21307 C03YHL 54583392 IC50 > 50000 nM T21307 C87ZTP 54583393 IC50 = 3100 nM T21307 C1E8RA 54583423 IC50 = 2000 nM T21307 C4ZX1L 54583424 IC50 = 14500 nM T21307 C32WCI 54583425 IC50 = 580 nM T21307 CL8ZK6 54583503 EC50 = 6.9 nM T21307 C0GZ2J 54583504 EC50 = 18 nM T21307 C3TSL4 54583881 EC50 = 10 nM T21307 CQ5Y3Z 54583882 EC50 = 11 nM T21307 CR9F5G 54584339 IC50 = 13000 nM T21307 CE7NU3 54584340 IC50 = 91000 nM T21307 CQ8T4Y 54584341 IC50 = 3200 nM T21307 CHE6X3 54584342 IC50 = 1900 nM T21307 CR0OA2 54584380 IC50 > 20000 nM T21307 C7D3UG 54584381 IC50 = 27000 nM T21307 C2JB8Y 54584382 IC50 = 150 nM T21307 CNB5A9 54584383 IC50 = 10000 nM T21307 CKR52F 54584384 IC50 = 2300 nM T21307 CX93NO 54584385 IC50 > 20000 nM T21307 C2U5RD 54584386 IC50 = 140 nM T21307 CCVF45 54584836 EC50 = 91 nM T21307 C4Z6HW 54585307 IC50 = 2500 nM T21307 C7YKL1 54585308 IC50 > 50000 nM T21307 CV4L9P 54585309 IC50 = 2300 nM T21307 CXY15G 54585310 IC50 > 50000 nM T21307 CS5PJ8 54585311 IC50 = 7000 nM T21307 C9ADW2 54585338 IC50 = 9300 nM T21307 C0QU1E 54585339 IC50 = 230 nM T21307 C4OXD2 54585340 IC50 = 1500 nM T21307 CNQ30S 54585341 IC50 = 30 nM T21307 C18HFD 54585792 EC50 = 15 nM T21307 C8E9PS 54585793 EC50 = 24 nM T21307 C5P0LQ 54585794 EC50 = 21 nM T21307 CG7OZ0 54585795 EC50 = 9.3 nM T21307 C89NVY 54585796 EC50 = 126 nM T21307 C09GHC 54586258 IC50 = 53000 nM T21307 CVW56O 54586259 IC50 = 35000 nM T21307 CC78LM 54586260 IC50 = 32000 nM T21307 C0NF4V 54586261 IC50 > 50000 nM T21307 CEDZ60 54586262 IC50 = 6900 nM T21307 CAU90X 54586298 IC50 = 460 nM T21307 CCI69U 54586299 IC50 = 1100 nM T21307 C74NWS 54586300 IC50 = 2500 nM T21307 C3CG1X 54586301 IC50 = 4300 nM T21307 C27JQM 54586302 IC50 = 1700 nM T21307 CI5OC9 54586303 IC50 = 13300 nM T21307 CRQ4V3 54586304 IC50 = 210 nM T21307 CPG54M 54586305 IC50 = 15000 nM T21307 C03UTH 54586306 IC50 = 27000 nM T21307 C7AVJ8 54586772 EC50 = 1.7 nM T21307 CJF8H2 54587285 IC50 = 13700 nM T21307 CFIB84 54587286 IC50 = 2700 nM T21307 CW2CN7 54587287 IC50 = 6900 nM T21307 CK06SU 54587326 IC50 = 2000 nM T21307 C3MZL4 54587327 IC50 = 11300 nM T21307 CJZ06G 54587328 IC50 = 40000 nM T21307 CA6T2C 54587329 IC50 = 940 nM T21307 C8BD9J 54587330 IC50 = 190 nM T21307 CVRT58 54587331 IC50 = 83 nM T21307 CW8G1C 54587411 EC50 = 288 nM T21307 CIF3X1 54587800 EC50 = 59 nM T21307 CX49CV 54587801 EC50 = 6.2 nM T21307 C5G7VA 54587802 EC50 = 6 nM T21307 C9ODN7 54694607 IC50 = 39000 nM T21307 C4OE1Z 54697518 IC50 = 130000 nM T21307 CE1ZK6 54759168 IC50 > 10000 nM T21307 C1XS2J 54760383 IC50 > 10000 nM T21307 C6ITG7 56659477 IC50 = 230 nM T21307 CB2V7L 56659478 IC50 = 8 nM T21307 CXR37P 56659479 IC50 = 900 nM T21307 CRQG79 56659480 IC50 = 4300 nM T21307 C16ENA 56659481 IC50 = 13 nM T21307 CX4LI2 56662940 IC50 = 80 nM T21307 CXL67Z 56662941 IC50 = 230 nM T21307 CX10VD 56662942 IC50 = 120 nM T21307 C0RDH6 56662943 IC50 = 4 nM T21307 CQ3MY5 56662944 IC50 = 6700 nM T21307 CPSO16 56666414 IC50 = 1200 nM T21307 CSLQ05 56666415 IC50 < 3 nM T21307 C9T1MD 56666416 IC50 < 3 nM T21307 CWP25J 56666417 IC50 = 20 nM T21307 CPUT19 56669830 IC50 = 140 nM T21307 CZO90M 56669831 IC50 < 3 nM T21307 C30ZLS 56669832 IC50 < 3 nM T21307 C1FCK8 56669833 IC50 = 4500 nM T21307 C16JTX 56669834 IC50 = 200 nM T21307 C02JLF 56669835 IC50 = 23 nM T21307 CB4ZI7 56673312 IC50 = 40 nM T21307 CN3W6Q 56673315 IC50 = 17 nM T21307 C6EHN5 56673316 IC50 < 3 nM T21307 CX0F9N 56673317 IC50 = 2500 nM T21307 C59QAE 56673318 IC50 = 120 nM T21307 CCR01T 56673319 IC50 = 34 nM T21307 C6HI1N 56676612 IC50 = 167 nM T21307 CYC71X 56676644 IC50 = 2700 nM T21307 C0XKE7 56676653 IC50 = 27 nM T21307 C4YS8L 56676654 IC50 < 3 nM T21307 CGPV75 56676655 IC50 < 3 nM T21307 CSEN25 56676656 IC50 < 3 nM T21307 C7N2VR 56676657 IC50 = 860 nM T21307 C40VTC 56676658 IC50 = 180 nM T21307 C3RDY2 56676664 IC50 = 73 nM T21307 C5GZ1O 56676665 IC50 = 85 nM T21307 C2T7JG 56679974 IC50 = 180 nM T21307 CE0R5T 56679977 IC50 = 175 nM T21307 CFM01T 56679978 IC50 = 230 nM T21307 C01DNE 56679979 IC50 = 1800 nM T21307 CV9I2X 56679980 IC50 = 3300 nM T21307 C1CQ6I 56683315 IC50 = 100 nM T21307 C71DPV 56683316 IC50 = 45 nM T21307 CT4E8R 56832546 IC50 = 16000 nM T21307 CBOD63 56835089 IC50 > 30000 nM T21307 CSD9L0 56835137 EC50 = 1 nM T21307 C0EL6D 56835138 EC50 = 2.3 nM T21307 CQ9VJ4 56835139 EC50 = 0.72 nM T21307 C0S9PV 56835140 EC50 = 2.6 nM T21307 C75FZB 56835141 EC50 = 1.1 nM T21307 C35LHC 56835142 EC50 = 2.5 nM T21307 C7NY9H 56835159 EC50 = 1.5 nM T21307 C1N9HR 56835160 EC50 = 2.7 nM T21307 CY5M7A 56950243 IC50 = 8 nM T21307 C1O2HA 56950796 IC50 = 2.9 nM T21307 C2F6QY 56950797 IC50 = 3.8 nM T21307 CET57W 57330141 EC50 = 170 nM T21307 CD50MC 57391312 IC50 = 128 nM T21307 CXN2L7 57391323 IC50 = 21 nM T21307 C4ZJN6 57391324 IC50 = 8 nM T21307 C56DCS 57391325 IC50 = 27 nM T21307 CO45NJ 57391326 IC50 = 52 nM T21307 CSZ40A 57391327 IC50 = 177 nM T21307 CH03RG 57391727 EC50 = 2.5 nM T21307 C4SJ8C 57392443 EC50 = 2100 nM T21307 C2JK9R 57392444 IC50 = 9.2 nM T21307 CLU61T 57392445 IC50 = 880 nM T21307 CVK8B2 57392446 IC50 = 18 nM T21307 CD1K5G 57393087 IC50 = 115 nM T21307 CPF7V3 57393088 IC50 = 10000 nM T21307 CKC94Q 57393102 IC50 = 285 nM T21307 COS70V 57393103 IC50 = 20 nM T21307 C02KUY 57393104 IC50 = 20 nM T21307 C3RV0Q 57393105 IC50 = 100 nM T21307 C9K7LA 57393461 EC50 = 1.4 nM T21307 C6U4RH 57393462 EC50 = 2.6 nM T21307 C79GXO 57393463 EC50 = 5.5 nM T21307 CH9A3E 57393464 EC50 = 5.1 nM T21307 CKM40Y 57393540 EC50 = 1.6 nM T21307 CC8XJ1 57394157 IC50 = 110 nM T21307 CFR1W7 57394816 IC50 = 9 nM T21307 C46XLG 57394830 IC50 = 24 nM T21307 CV4AJ5 57394831 IC50 = 258 nM T21307 CD6Y9Z 57395116 IC50 > 30000 nM T21307 C8W6IG 57395117 IC50 > 30000 nM T21307 CT5K2B 57395185 EC50 = 3.3 nM T21307 CVU6D5 57395186 EC50 = 1.9 nM T21307 CD8YA1 57395255 EC50 = 3.1 nM T21307 CN7OK0 57395930 IC50 = 258 nM T21307 CHP9A3 57395938 EC50 = 1500 nM T21307 C9OBF4 57395939 IC50 = 15 nM T21307 C5Q1MJ 57396580 IC50 = 12 nM T21307 CG7S0D 57396882 IC50 > 30000 nM T21307 C5TQ0F 57396965 EC50 = 1.3 nM T21307 CS34UH 57396966 EC50 = 4.1 nM T21307 CXK4C5 57398359 IC50 = 1450 nM T21307 C1LT5B 57398374 IC50 = 14 nM T21307 CK4E3V 57398375 IC50 = 12 nM T21307 CTDC86 57398376 IC50 = 9 nM T21307 C6HEN3 57398709 EC50 = 4.2 nM T21307 C2TLU4 57398710 EC50 = 1.6 nM T21307 CPF4Z6 57400015 IC50 = 10000 nM T21307 CMZ7G6 57400017 IC50 = 1920 nM T21307 C6Q4AR 57400031 IC50 = 19 nM T21307 CLU48P 57400032 IC50 = 43 nM T21307 CETO45 57400383 EC50 = 2.4 nM T21307 CK1JD6 57400384 EC50 = 11 nM T21307 CXES59 57400385 EC50 = 9.1 nM T21307 C4RV5D 57400386 EC50 = 0.71 nM T21307 CLVA04 57400468 EC50 = 5.1 nM T21307 C0UDY9 57401151 EC50 = 2000 nM T21307 CO5SV2 57401826 IC50 = 79 nM T21307 CO0D5A 57401827 IC50 = 41 nM T21307 CC4FR2 57401828 IC50 = 12 nM T21307 C8GD3E 57401829 IC50 = 110 nM T21307 C6GW3V 57401844 IC50 = 12 nM T21307 CCI37Z 57402183 EC50 = 0.62 nM T21307 CE20RY 57402270 EC50 = 14 nM T21307 C19MQN 57402271 EC50 = 15 nM T21307 C5X8GD 57402272 EC50 = 1.6 nM T21307 C8IY0J 57403532 IC50 = 4743 nM T21307 CLA50Z 57403533 IC50 = 70 nM T21307 CYTK68 57403552 IC50 = 9 nM T21307 CQ2X7V 57403940 EC50 = 2.5 nM T21307 CWIA09 57403941 EC50 = 6.2 nM T21307 CPY13B 57404001 EC50 = 0.96 nM T21307 C48ATX 57752723 IC50 = 650 nM T21307 CJVG28 57753017 IC50 = 26000 nM T21307 CXJ63M 59603829 IC50 > 100000 nM T21307 CQEU96 59603842 IC50 = 390 nM T21307 C1MR8Q 60097495 IC50 > 1000 nM T21307 CH1SL5 60199603 IC50 > 300000 nM T21307 CM4RV5 60199605 IC50 > 300000 nM T21307 CJHP90 60199775 IC50 > 100000 nM T21307 CTA0Q3 60199933 IC50 = 2000 nM T21307 CJR74L 60199934 IC50 > 100000 nM T21307 CCO6P4 60199938 IC50 > 100000 nM T21307 CBJ6W4 60199940 IC50 > 100000 nM T21307 C6FY5G 60199942 IC50 = 25000 nM T21307 CK4Z0H 60200097 IC50 = 400 nM T21307 CZ34FG 60200098 IC50 > 100000 nM T21307 CWQN93 60200099 IC50 > 100000 nM T21307 CYP57O 60200105 IC50 = 89000 nM T21307 C8G2DO 60200252 IC50 = 2500 nM T21307 C08IER 60200253 IC50 = 8700 nM T21307 CY7I8R 60200254 IC50 = 4100 nM T21307 CN42BP 60200255 IC50 = 83000 nM T21307 CCON02 60200403 IC50 = 510 nM T21307 CLW75Z 60200406 IC50 > 300000 nM T21307 CV8X3M 60200408 IC50 = 1200 nM T21307 CD6E5Q 60200569 IC50 = 700 nM T21307 C49KDS 60200570 IC50 = 700 nM T21307 C5E9MC 60200571 IC50 = 1400 nM T21307 C2O9KV 60200572 IC50 = 1900 nM T21307 CLVK19 60200736 IC50 = 3000 nM T21307 CH59YJ 60200737 IC50 = 130 nM T21307 CCG75S 60200900 IC50 = 160 nM T21307 CC4V6R 60200902 IC50 = 140 nM T21307 CG47WK 60200904 IC50 = 57 nM T21307 CF7M2W 60200906 IC50 = 76 nM T21307 CN9GQ8 60201066 IC50 = 54 nM T21307 CRN3D6 60201068 IC50 = 200 nM T21307 C1ER6C 60201070 IC50 = 1700 nM T21307 CR3AJ9 60201072 IC50 = 1500 nM T21307 C1HSE0 67035086 IC50 > 10000 nM T21307 CWI6K5 67035106 IC50 > 10000 nM T21307 C38RGB 67035556 IC50 > 10000 nM T21307 CV63UL 67240318 IC50 > 10000 nM T21307 C8I7GC 68293638 IC50 > 10000 nM T21307 CD56XK 68293660 IC50 > 10000 nM T21307 C5DGR9 69036886 IC50 = 10000 nM T21307 C4NIQ0 70681191 EC50 = 5000 nM T21307 CMW54H 70681757 IC50 = 50 nM T21307 CV71DA 70681758 IC50 = 60 nM T21307 C7Z9NI 70681765 IC50 = 160 nM T21307 C39HGR 70681766 IC50 = 790 nM T21307 CKH75E 70681767 IC50 > 10000 nM T21307 C8N7ZA 70683279 IC50 > 20000 nM T21307 C74GUS 70683871 IC50 = 3700 nM T21307 CVC7Z9 70683872 EC50 = 3700 nM T21307 CXR08J 70683873 IC50 = 70 nM T21307 C5V3YS 70683880 IC50 = 1200 nM T21307 C32BTE 70683881 IC50 = 330 nM T21307 C8SO1U 70683882 IC50 = 480 nM T21307 C76YMN 70683883 IC50 = 50 nM T21307 CO1K9V 70685385 EC50 > 8000 nM T21307 CG1S9H 70685386 EC50 > 3400 nM T21307 C8U6CW 70685387 EC50 = 900 nM T21307 CL40AD 70685388 IC50 = 1200 nM T21307 CNS08W 70686009 EC50 = 6700 nM T21307 C4FW2I 70686016 IC50 = 100 nM T21307 C1ODL9 70686017 IC50 = 970 nM T21307 CMWO17 70686018 IC50 = 310 nM T21307 COK08M 70686019 IC50 = 5300 nM T21307 CR2J5T 70686020 IC50 = 190 nM T21307 CUT6Y4 70687520 EC50 = 1600 nM T21307 CNGO72 70687521 EC50 > 8000 nM T21307 C1EB3T 70687522 EC50 = 4000 nM T21307 CCR0X9 70688136 IC50 > 10000 nM T21307 C0EF8I 70688137 IC50 = 6200 nM T21307 C71ZLE 70688146 EC50 = 820 nM T21307 CPUK45 70688147 IC50 = 1300 nM T21307 CWQF14 70689580 EC50 = 8000 nM T21307 C1SAT7 70689581 IC50 = 6900 nM T21307 CHV9E1 70689582 EC50 = 1900 nM T21307 CP5E3M 70689583 EC50 = 9000 nM T21307 C6JX3G 70689597 EC50 = 530 nM T21307 CN2HL7 70690181 IC50 = 180 nM T21307 CE49NM 70691708 EC50 > 5000 nM T21307 CXW2E9 70691709 EC50 = 1400 nM T21307 CDN98S 70691710 IC50 = 20000 nM T21307 CI1JX3 70691711 EC50 = 1300 nM T21307 CA19OU 70691712 IC50 = 650 nM T21307 C8XIW3 70691713 IC50 = 440 nM T21307 C86IAB 70692321 IC50 = 110 nM T21307 CBG9Z2 70692322 EC50 = 3000 nM T21307 CG43UY 70692323 EC50 = 2700 nM T21307 CF40ZY 70692331 IC50 = 70 nM T21307 CNH5Z1 70692332 IC50 > 10000 nM T21307 C2LR5S 70692333 IC50 > 10000 nM T21307 C0KL9A 70693786 IC50 = 15000 nM T21307 C3XWI6 70694383 IC50 = 3400 nM T21307 C1CZ7X 70694393 IC50 = 190 nM T21307 CQ1SL7 70694394 EC50 = 730 nM T21307 CZ42MX 70694395 IC50 = 220 nM T21307 CB6GL8 70695897 EC50 = 3900 nM T21307 CA0XD9 70695898 IC50 = 130 nM T21307 CA59LE 70696462 IC50 = 1400 nM T21307 CDU7Z4 70696464 IC50 = 380 nM T21307 CH0B8N 70789756 IC50 > 30000 nM T21307 C91HPI 71300299 IC50 > 5000 nM T21307 C8FG2N 71453355 IC50 = 12000 nM T21307 CH8B6T 71460534 IC50 = 7000 nM T21307 CWJS14 71462243 IC50 = 11000 nM T21307 CXP0Q8 71462244 IC50 > 100000 nM T21307 CCN01X 71547862 IC50 > 10000 nM T21307 CA3O6K 71552696 IC50 > 30000 nM T21307 C1NPL0 71552941 IC50 > 30000 nM T21307 CA4PS8 71552942 IC50 > 30000 nM T21307 C3UA9C 71553011 IC50 = 30000 nM T21307 CEZ15Y 71553012 IC50 = 30000 nM T21307 CVIA91 71553085 IC50 = 30000 nM T21307 C1TR3O 71553152 IC50 = 30000 nM T21307 C08XIE 71614291 IC50 = 4000 nM T21307 C7J2KQ 71614497 IC50 = 1980 nM T21307 C79AHD 71625453 IC50 = 12 nM T21307 CGBD78 71625454 IC50 = 74 nM T21307 C34FMK 71625455 IC50 = 14 nM T21307 CLJC80 71625566 IC50 = 4.9 nM T21307 C2C5ZN 71625567 IC50 = 21 nM T21307 C7CFY6 71625568 IC50 = 8.4 nM T21307 CD9QN2 71625569 IC50 = 6.8 nM T21307 C5NPI8 71625570 IC50 = 28 nM T21307 CC2LO7 71625683 IC50 = 3 nM T21307 C4IE1T 71625684 IC50 = 8.9 nM T21307 CXSI14 71718330 IC50 > 100000 nM T21307 C1TM3P 71720141 IC50 > 100000 nM T21307 CB8ZU1 72188683 IC50 = 840 nM T21307 C1HW4B 89735655 IC50 = 7800 nM T21307 CY0UC4 90645194 IC50 > 10000 nM T21307 C0Y8ZK 91933875 IC50 > 1000 nM T21307 CAU45T 91971978 IC50 = 25.5 nM T21307 CY7BI2 118706214 IC50 > 10000 nM T21307 CRE9N3 118707413 IC50 = 84.7 nM T21307 C9CXM8 118707414 IC50 = 14.3 nM T21307 CZ27VM 118707415 IC50 = 23.3 nM T21307 CJ7H5V 118707416 IC50 = 157 nM T21307 C6ZUW0 118707417 IC50 = 450.1 nM T21307 CX9CQ6 118707418 IC50 = 95.4 nM T21307 C1MU8J 118707419 IC50 = 16.2 nM T21307 C9SC5K 118707420 IC50 = 13 nM T21307 C5KNV1 118707421 IC50 = 17.4 nM T21307 CZ8WX0 118707422 IC50 = 22.3 nM T21307 C4LGD3 118707423 IC50 = 31.3 nM T21307 C4Z7CP 118707424 IC50 = 43.5 nM T21307 CS9IE1 118707425 IC50 = 7.7 nM T21307 CIHD60 118707426 IC50 = 35.7 nM T21307 CT5M1E 118707427 IC50 = 36.7 nM T21307 CFD8B6 118707428 IC50 = 26 nM T21307 C4QNO9 118707429 IC50 = 160 nM T21307 CI56JD 118707430 IC50 = 3730 nM T21307 CP5CT4 118708080 IC50 = 3390 nM T21307 C5ET8O 118708081 IC50 = 65 nM T21307 CF6C9Y 118708082 IC50 = 55.3 nM T21307 CN5HT9 118708083 IC50 = 74.9 nM T21307 C6VJG2 118708084 IC50 = 66.5 nM T21307 CO85DL 118708085 IC50 = 25.8 nM T21307 CO63YL 118708086 IC50 = 24.9 nM T21307 C85PUD 118708087 IC50 = 26 nM T21307 C7T8ML 122193924 IC50 = 4200 nM T21307 CI76XH 122193925 IC50 = 3600 nM T21307 COJ8E0 122193926 IC50 = 26000 nM T21307 CD1B3O 122193927 IC50 = 27000 nM T21307 C12RNT 122194063 IC50 = 31000 nM T21307 C5VLM4 122194064 IC50 = 3300 nM T21307 CB9X2N 122194065 IC50 = 1700 nM T21307 CF29KI 122194066 IC50 = 6900 nM T21307 CV7FU1 122194067 IC50 > 40000 nM T21307 CCEO60 122194068 IC50 = 36000 nM T21307 CEL6W8 122194069 IC50 = 7800 nM T21307 C47LMR 122194070 IC50 = 2400 nM T21307 CXGZ75 122194071 IC50 = 1900 nM T21307 CFC1H8 122194072 IC50 = 10000 nM T21307 CKQ6T0 122194073 IC50 = 8000 nM T21307 C61CHY 122194074 IC50 > 20000 nM T21307 CKQD39 122194075 IC50 > 20000 nM T21307 C1GD5P 122194203 IC50 = 32000 nM T21307 CJO53H 122194204 IC50 = 4500 nM T21307 CA07QN 122194205 IC50 = 2200 nM T21307 CXKS58 122194206 IC50 = 750 nM T21307 C1LJH0 122194207 IC50 = 6700 nM T21307 C5Z1KF 122194208 IC50 = 11000 nM T21307 C4O1FD 122194209 IC50 = 19000 nM T21307 C0EL5F 122194210 IC50 = 11800 nM T21307 CI2EU6 122194211 IC50 = 8000 nM T21307 C8J7AZ 122194212 IC50 = 20000 nM T21307 CTQ81J 122194213 IC50 = 19000 nM T21307 CS40VC 122194214 IC50 = 16200 nM T21307 C6DE2B 122194215 IC50 = 14500 nM T21307 C69ISU 122197365 IC50 = 180 nM T21307 CMQY01 122197366 IC50 = 470 nM T21307 C29IEJ 122197367 IC50 = 403 nM T21307 CS3C7H 122197368 IC50 = 419 nM T21307 C0GP7A 122197369 IC50 = 64800 nM T21307 CAE09S 122197370 IC50 = 460 nM T21307 CY3D7O 122197371 IC50 > 200000 nM T21307 CXZK31 122197372 IC50 = 490 nM T21307 C9O0XD 122197373 IC50 = 530 nM T21307 CD9UN3 122197374 IC50 = 560 nM T21307 CC4R2V 122197375 IC50 = 620 nM T21307 CIU36T 122197376 IC50 = 690 nM T21307 CLW25T 122197377 IC50 = 770 nM T21307 CM0E1X 122197378 IC50 = 850 nM T21307 CYO0W5 122197379 IC50 > 200000 nM T21307 CO8S7G 122197380 IC50 = 130 nM T21307 CL6I1R 122197381 IC50 = 1680 nM T21307 CM05IY 122197382 IC50 = 237 nM T21307 C59IZO 122197383 IC50 = 6180 nM T21307 C3AN7Z 122197384 IC50 = 4220 nM T21307 CT4N8D 122197385 IC50 > 200000 nM T21307 CTG74O 122197386 IC50 = 1940 nM T21307 COGP03 122197387 IC50 = 12800 nM T21307 CLA4C3 127043567 IC50 = 22000 nM T21307 C7TPU9 127043735 IC50 = 740 nM T21307 C86ZUT 127044221 IC50 = 5800 nM T21307 C0FM1R 130196825 IC50 > 30000 nM T21307 CUO0C5 132156633 IC50 > 10000 nM T21307 CKHI48 135441367 IC50 = 170 nM T21307 CTJ48K 135524085 IC50 = 82 nM T21307 CVI72G 135524105 IC50 = 1300 nM T21307 CN3A6B 135524106 IC50 = 290 nM T21307 CFB3N6 135524107 IC50 = 1700 nM T21307 CJM1T4 135524108 IC50 = 150 nM T21307 CGE3H6 135524110 IC50 = 42 nM T21307 CHIJ03 135524114 IC50 = 1230 nM T21307 C28JET 135524115 IC50 = 350 nM T21307 C5T0XB 135524116 IC50 = 1450 nM T21307 CNIJ80 135524117 IC50 = 200 nM T21307 CEKL94 135524133 IC50 = 1260 nM T21307 CRT39X 135524134 IC50 = 340 nM T21307 CUT1W7 135524168 IC50 = 51 nM T21307 C45RIY 135556284 IC50 = 410 nM T21307 COCR58 135556294 IC50 = 21 nM T21307 CEK31P 135566415 IC50 > 20000 nM T21307 CRJ45X 135589980 IC50 > 50000 nM T21307 C6MX9S 135797231 IC50 = 14 nM T21307 CX4ZB3 135863110 IC50 = 19000 nM T21307 CX5E9C 135874060 IC50 = 540 nM T21307 CU0SO9 135874061 IC50 = 5200 nM T21307 CP3LQ9 135890414 IC50 = 10 nM T21307 CXV1Y5 135890416 IC50 = 25 nM T21307 CZ5UN7 135890420 IC50 = 116 nM T21307 CL6AO7 135890427 IC50 = 1189 nM T21307 CV3E0X 135890430 IC50 = 8 nM T21307 C0OM5P 135890431 IC50 = 10 nM T21307 CP1Y5C 135890437 IC50 = 253 nM T21307 CH26QS 135890446 IC50 = 5 nM T21307 C5RPY8 135971385 IC50 = 160 nM T21307 CHA4N2 136013680 IC50 > 10 nM T21307 C6T3QE 136025993 IC50 = 172 nM T21307 C5XIE8 136026041 IC50 = 35000 nM T21307 C6V5FC 136079665 IC50 = 1 nM T21307 C49DYH 136079673 IC50 = 60 nM T21307 CX05YU 136099796 IC50 = 190 nM T21307 C1YUD0 136219394 IC50 > 10 nM T21307 CIU8W3 136254389 IC50 > 10 nM T21307 C8GQD5 137636872 IC50 > 10000 nM T21307 C9Y4DC 138978963 IC50 < 3 nM T21307 CZ2XH5 139187793 IC50 = 2300 nM T21307 C6VB3O 145925651 IC50 >= 5000 nM T21307 CJXP51 145979306 IC50 < 3 nM T21307 C3ELP8 145989661 IC50 < 3 nM T21307 D00ERW 44444843 Ki = 3886 nM T21307 D00HVA 11624601 Ki > 8400 nM T21307 D00TBD 10461815 IC50 > 10000 nM T21307 D01YWE 25207521 IC50 = 390 nM T21307 D03DZO 11715767 IC50 = 470 nM T21307 D03MUZ 17759555 IC50 = 40200 nM T21307 D06HVH 54613583 IC50 > 10000 nM T21307 D06KSF 9549300 IC50 = 110000 nM T21307 D06QBJ 44631903 Ki = 5 nM T21307 D06WGX 9549184 IC50 > 25000 nM T21307 D08HFG 24809764 IC50 > 10000 nM T21307 D09HVH 135566652 IC50 > 10 nM T21307 D0CM6T 11314340 Ki = 1100 nM T21307 D0D6DH 10125830 IC50 > 50000 nM T21307 D0D6MH 11617559 IC50 > 10000 nM T21307 D0E3OL 4567175 IC50 > 200000 nM T21307 D0EW9J 10389239 EC50 = 49 nM T21307 D0F0AU 44405988 IC50 > 20000 nM T21307 D0O6OH 71553154 IC50 = 18570 nM T21307 D0O7UT 11382492 Ki = 330 nM T21307 D0Q3NG 11715520 Ki > 8400 nM T21307 D0S7IE 11658882 Ki > 8400 nM T21307 D0T8NU 16757525 IC50 = 510 nM T00302 D00EPS 449051 Ki = 78 nM T00302 C4RSI0 46899736 Ki = 108 nM T00302 CLC94G 46918674 Ki = 54.3 nM T00302 C54AGL 46918753 Ki = 112.3 nM T00302 CU1DK9 49835415 Ki = 40 nM T00302 C8NZ1B 49835505 Ki = 430 nM T00302 CGXJ39 49835506 Ki = 51 nM T00302 CIB2S3 49835507 Ki = 98 nM T00302 CA30SZ 49835508 Ki = 63 nM T00302 C17XIQ 49835556 Ki = 53 nM T00302 C0OQ8N 49835557 Ki = 13 nM T00302 C03HXU 49835559 Ki = 311 nM T00302 CCJ92X 49835606 Ki = 168 nM T00302 CB08CW 53379392 Ki = 17 nM T00302 CZ39YM 56659848 Ki = 135 nM T00302 CH3J4I 56659849 Ki = 149 nM T00302 CA32CM 56659850 Ki = 30 nM T00302 CFY8L6 56659851 Ki = 57 nM T00302 CK7J8U 56659852 Ki = 422 nM T00302 CDY0G4 56663317 Ki = 158 nM T00302 CPG61H 56663318 Ki = 221 nM T00302 CKO4M6 56663319 Ki = 15 nM T00302 C1M0YS 56666743 Ki = 73 nM T00302 C6EU5O 56666744 Ki = 210 nM T00302 CNYB70 56666745 Ki = 34 nM T00302 CC3D4Z 56666746 Ki = 47 nM T00302 CCM80T 56670171 Ki = 36 nM T00302 C8ESB6 56673691 Ki = 76 nM T00302 CXGO13 56673692 Ki = 120 nM T00302 CDS6E7 56673693 Ki = 1425 nM T00302 CGM2J4 56673694 Ki = 22 nM T00302 C4T6NO 56673695 Ki = 34 nM T00302 CRD28L 56673696 Ki = 512 nM T00302 C4DB5K 56677005 Ki = 38 nM T00302 C1TH3W 56677006 Ki = 68 nM T00302 CY34VE 56677007 Ki = 14 nM T00302 CSW9I3 56677008 Ki = 23 nM T00302 C72IHP 56680339 Ki = 38 nM T00302 CWE25P 56683657 Ki = 43 nM T00302 CVR5F7 56683658 Ki = 183 nM T00302 CV06WG 56683659 Ki = 202 nM T00302 C1OJW0 56683660 Ki = 457 nM T00302 D07ZRG 46899577 Ki = 19 nM T00302 D0W2SV 70689167 Ki = 8.4 nM T01148 D0G5UB 2161 IC50 = 851.14 nM T01148 D0OB0F 5328940 IC50 = 471 nM T01148 D02XNW 5494449 IC50 = 6.22 nM T01148 D09JEJ 24748573 IC50 = 35 nM T01148 D0E3TC 44259 IC50 = 2.18 nM T01148 D03BNU 59604787 IC50 > 10000 nM T01148 D09FGW 56646218 IC50 = 1 nM T01148 D0T3ME 156422 IC50 > 30000 nM T01148 CJ2T3N 10023121 IC50 = 383 nM T01148 C0IVL9 10347359 IC50 = 6 nM T01148 CW5C9X 11186250 IC50 > 3162.28 nM T01148 CM21YJ 11453049 IC50 > 3162.28 nM T01148 CACS26 11561968 Ki > 2000 nM T01148 CGX96V 11626927 IC50 = 72 nM T01148 CJ9KN7 11683817 IC50 > 10000 nM T01148 CU0E8O 11690457 Ki > 2000 nM T01148 CB0AP2 11705863 Ki > 10000 nM T01148 CM7S0Z 12852146 IC50 = 400 nM T01148 C41KUL 15571856 IC50 = 524.81 nM T01148 C5VPH9 16129448 IC50 = 1070 nM T01148 C7YG1N 24759534 IC50 < 10 nM T01148 CLBP72 24798571 IC50 > 4000 nM T01148 CU19EF 44231127 IC50 = 8 nM T01148 CI3BA2 44462961 IC50 = 820 nM T01148 C3XY7U 44464266 IC50 = 11 nM T01148 CQ8BA1 44464268 IC50 = 3 nM T01148 CLI16E 44465026 IC50 = 8 nM T01148 C6RXW1 44465027 IC50 = 9 nM T01148 C8CF6N 44465029 IC50 = 3200 nM T01148 CEK2D3 44465285 IC50 = 4 nM T01148 C6M9IQ 44465820 IC50 = 2 nM T01148 CJW93H 44466599 IC50 = 28 nM T01148 C3VRO9 44557921 IC50 > 10000 nM T01148 CEQN27 52936621 Ki > 1000 nM T01148 C8NA4L 53384644 IC50 > 30000 nM T01148 C03XBT 57328467 EC50 = 139 nM T01148 CXJ35L 57328543 EC50 = 35 nM T01148 CCF61V 57328544 EC50 = 34 nM T01148 C39KXI 57328545 EC50 = 17 nM T01148 C2TC6M 59225246 IC50 = 63 nM T01148 C8K5QN 59225250 IC50 = 6 nM T01148 CT70FI 59225251 IC50 = 2 nM T01148 COCB23 59225272 IC50 = 7 nM T01148 CAK48J 59225283 IC50 = 16 nM T01148 CH0G1X 59225285 IC50 = 15 nM T01148 C1W9GK 59225297 IC50 = 3 nM T01148 C3SBA4 59225303 IC50 = 8 nM T01148 C8TQB4 59225307 IC50 > 1000 nM T01148 CT5OV9 59225334 IC50 = 13 nM T01148 CHV18S 59225349 IC50 = 9 nM T01148 C7FQD2 59225366 IC50 = 110 nM T01148 CM48WR 59225375 IC50 = 2 nM T01148 CXJC43 59225411 IC50 = 2 nM T01148 C4K7PD 59225430 IC50 > 1000 nM T01148 CXJ63M 59603829 IC50 < 10 nM T01148 CQEU96 59603842 IC50 < 1 nM T01148 COH62U 60097413 IC50 > 10000 nM T01148 C1MR8Q 60097495 IC50 > 1000 nM T01148 C37NKO 67129970 IC50 > 10000 nM T01148 CK80LJ 67130050 IC50 > 10000 nM T01148 CV63UL 67240318 IC50 > 10000 nM T01148 C7GRV2 68755406 IC50 > 10000 nM T01148 C5DGR9 69036886 IC50 = 10000 nM T01148 C6F4QX 70681026 IC50 = 151 nM T01148 CQ63HX 70681027 IC50 = 231 nM T01148 CR2QO7 70681028 IC50 = 106 nM T01148 CRZ36H 70681029 IC50 = 12000 nM T01148 CZ4OY5 70681030 IC50 = 8 nM T01148 CU6NE9 70681031 IC50 = 59 nM T01148 CPOV92 70681032 IC50 = 3 nM T01148 COHI26 70681033 EC50 = 12 nM T01148 C48POI 70683150 IC50 = 468 nM T01148 C25FGR 70683151 IC50 = 345 nM T01148 CSN7L4 70683152 IC50 = 178 nM T01148 C6XO5Q 70683153 IC50 = 288 nM T01148 CW8LF0 70683154 IC50 = 1520 nM T01148 C7EH1D 70683155 EC50 = 11 nM T01148 C5I7DW 70685226 IC50 = 426 nM T01148 COYD53 70685227 IC50 = 2740 nM T01148 CU47OG 70685228 IC50 = 257 nM T01148 CZ6NH0 70685229 IC50 = 388 nM T01148 CE65KV 70685230 IC50 = 213 nM T01148 CRK92N 70685231 EC50 = 14 nM T01148 CA57VF 70685232 EC50 = 26 nM T01148 CID9O3 70685233 IC50 = 4 nM T01148 CN2O6T 70687384 IC50 = 229 nM T01148 C4Q5MO 70687385 IC50 = 196 nM T01148 CA0FE8 70687386 EC50 = 111 nM T01148 CQH9A0 70687387 EC50 = 73 nM T01148 CMA7J1 70687388 EC50 = 6 nM T01148 CWD19I 70689442 IC50 = 2290 nM T01148 CW9O7S 70689443 IC50 = 105 nM T01148 CS7LM1 70689444 IC50 = 65 nM T01148 C1MSF8 70689445 IC50 = 233 nM T01148 CD5V2S 70689446 IC50 = 162 nM T01148 CEGM27 70689447 EC50 = 20 nM T01148 C80CWD 70689448 EC50 = 8 nM T01148 CQ1X4K 70691555 IC50 = 335 nM T01148 CN15SY 70691556 IC50 = 4 nM T01148 CO9KZ3 70693645 IC50 = 9550 nM T01148 CG9PD4 70695751 IC50 = 1220 nM T01148 C0B7XU 70695752 IC50 = 10300 nM T01148 CC6ZN8 70695753 IC50 = 1410 nM T01148 CP3G9T 70695755 IC50 = 111 nM T01148 CH2YA1 70695756 IC50 = 93 nM T01148 C47HZW 70695757 IC50 = 192 nM T01148 CL71AV 70695758 IC50 = 39 nM T01148 C2EI9Z 70695759 EC50 = 25 nM T01148 CZ4W6K 70695760 EC50 = 84 nM T01148 CS37NT 71450663 IC50 = 22 nM T01148 CF4P1N 71450664 IC50 > 10000 nM T01148 C2NCX1 71450665 IC50 = 7 nM T01148 CB9H5Y 71450666 IC50 = 7 nM T01148 CO7M9X 71452497 IC50 > 1000 nM T01148 C9I5GF 71454257 IC50 = 3600 nM T01148 C8OWL6 71456015 IC50 = 8 nM T01148 C4QUL2 71456016 IC50 = 450 nM T01148 C6E7MH 71457819 IC50 = 4300 nM T01148 CID65O 71459725 IC50 = 430 nM T01148 CYL46C 71459726 IC50 = 7 nM T01148 CD1W8C 71459727 IC50 = 4 nM T01148 CH83WB 71461445 IC50 = 10 nM T01148 CYN6R5 71461446 IC50 = 9 nM T01148 CET01R 71463176 IC50 = 560 nM T01148 CE9UA2 71463177 IC50 > 10000 nM T01148 C75RVU 71463178 IC50 = 60 nM T01148 C0DL3F 72698602 IC50 < 1 nM T01148 C42MXW 76310923 IC50 = 46 nM T01148 C0MR6F 76310924 IC50 = 136 nM T01148 CJ3I5E 76310925 IC50 = 1040 nM T01148 C6EI1G 76310926 IC50 = 256 nM T01148 CVP8Z4 76310927 IC50 = 129 nM T01148 C9MG7U 76314564 IC50 = 78 nM T01148 CU8EW0 76318141 IC50 = 759 nM T01148 C80VJZ 76318142 IC50 = 98 nM T01148 C6ZOM5 76321826 IC50 = 37 nM T01148 C5MRE6 76321827 IC50 = 268 nM T01148 CZ0XB7 76321828 IC50 = 1050 nM T01148 C1BJ5I 76321829 IC50 > 30000 nM T01148 C8Z6XR 76325460 IC50 = 2170 nM T01148 CKZ4F9 76325461 IC50 = 460 nM T01148 CTA86L 76325462 IC50 = 89 nM T01148 C9B2NA 76325463 IC50 = 859 nM T01148 CLF2S7 76325464 IC50 = 1800 nM T01148 CI7WT3 76325465 IC50 = 49 nM T01148 CT1R6E 76329005 IC50 = 7 nM T01148 CT4FE5 76329006 IC50 = 650 nM T01148 C8ZTP6 76332688 IC50 = 203 nM T01148 C0PRE8 76336290 IC50 = 128 nM T01148 CF1JW0 76336291 IC50 = 30 nM T01148 C1HW4B 89735655 IC50 < 10 nM T01148 CC23OD 91970516 IC50 = 0.06 nM T01148 CQCX41 118737057 IC50 > 10000 nM T01148 CTW92Q 121230617 IC50 = 13 nM T01148 CZ71IR 124108661 IC50 = 1.3 nM T01148 CWS5C4 129245211 IC50 = 372 nM T01148 CH91ON 129245363 IC50 = 9 nM T01148 C6A1LP 129245450 IC50 = 273 nM T01148 COKE50 129245476 IC50 = 764 nM T01148 CA2N5C 129245517 IC50 = 50 nM T01148 C0E2RU 129245526 IC50 = 2270 nM T01148 C9J8HZ 129245530 IC50 = 148 nM T01148 C52PNC 129245623 IC50 = 391 nM T01148 CL21HY 129245681 IC50 = 115 nM T01148 C1QKC7 129245769 IC50 = 34 nM T01148 CEYK58 129245795 IC50 = 5 nM T01148 CFP0G6 129245828 IC50 = 2490 nM T01148 COR37Y 129245842 IC50 = 72 nM T01148 CKB5C8 129245918 IC50 = 58 nM T01148 CQJK71 129246093 IC50 = 2 nM T01148 C0GC7N 129246130 IC50 = 55 nM T01148 C09MDW 129260549 IC50 = 2660 nM T01148 CCF8W2 129261617 IC50 = 10 nM T01148 CG5O2J 129261641 IC50 = 15 nM T01148 CPEA28 130275058 IC50 = 2300 nM T01148 C1BPS0 130275075 IC50 = 290 nM T01148 CSQ0O5 130275093 IC50 = 760 nM T01148 CS8YR1 130275108 IC50 = 550 nM T01148 CCWF83 130275116 IC50 = 300 nM T01148 CJ4GK2 130275332 IC50 = 630957.34 nM T01148 CYHA01 130275488 IC50 = 2290.87 nM T01148 CAT2Q7 130275498 IC50 = 1700 nM T01148 C7S0KD 130275500 IC50 = 1800 nM T01148 CU8IR7 130275554 IC50 = 4600 nM T01148 C6GSW1 130276189 IC50 = 570 nM T01148 C6HY7G 130276200 IC50 = 524807.46 nM T01148 C9G2SC 130276225 IC50 = 750 nM T01148 C7NCV5 130276229 IC50 = 270 nM T01148 CZ9K7R 130276230 IC50 = 830 nM T01148 CD6QO8 130276741 IC50 = 860 nM T01148 CR43KG 130276782 IC50 = 830 nM T01148 CS16TD 130276801 IC50 = 398.11 nM T01148 C1NWB5 130276805 IC50 = 490 nM T01148 CJ2T7Z 130276806 IC50 = 1900 nM T01148 CAQ89B 130276808 IC50 = 750 nM T01148 C90IYP 130276898 IC50 = 12000 nM T01148 COA70I 130276966 IC50 = 790 nM T01148 CPAX52 130276970 IC50 = 440 nM T01148 C8M6VS 130289650 IC50 = 537.03 nM T01148 C1NL4U 130290291 IC50 = 1900 nM T01148 CM65GQ 130290300 IC50 = 1300 nM T01148 CV0TH9 132000066 EC50 = 53900 nM T01148 C5UOY0 136266076 IC50 = 201 nM T01148 C8KJ9Z 137479135 IC50 = 1140 nM T01148 CVHF30 137479140 IC50 = 388 nM T01148 C7B4NR 137479154 IC50 = 5070 nM T01148 CO3NT9 137553174 IC50 = 1000 nM T01148 CI1E8V 137634241 IC50 = 7610 nM T01148 CM07EU 145714274 IC50 = 1 nM T01148 C9ISH6 145925685 IC50 = 30 nM T01148 C1A3HL 145988072 IC50 = 489.78 nM T01148 CT4M9E 145989247 IC50 = 1096.48 nM T01148 C7CH9V 146014951 IC50 = 2 nM T01148 CJB1R5 155511461 IC50 = 2 nM T01148 CV36FS 155512885 IC50 = 188 nM T01148 C2MD1Q 155513187 IC50 > 10000 nM T01148 C80CTM 155520004 IC50 = 1210 nM T01148 CZ0WO7 155523990 IC50 = 2 nM T01148 CHMV49 155525041 IC50 = 93 nM T01148 C82MLZ 155526827 IC50 = 29 nM T01148 CK2RM8 155528214 IC50 = 16700 nM T01148 CH0S4T 155530766 IC50 < 100 nM T01148 C8O6WA 155542495 IC50 = 1060 nM T01148 CHD09S 155543566 IC50 = 7 nM T01148 C2Y4AG 155546383 IC50 = 5 nM T01148 C6JWS0 155560801 IC50 = 281 nM T01148 CQRO74 155567366 IC50 = 98 nM T01148 D00ERW 44444843 Ki > 1525 nM T01148 D03BJF 44465558 IC50 = 6 nM T01148 D06ZIO 44464263 IC50 = 19 nM T01148 D0J3LR 11634725 Ki > 10000 nM T01148 D0RG0Z 10077147 IC50 = 6 nM T66383 D0C9MA 118323590 IC50 = 4 nM T66383 D01IBO 9822205 IC50 = 96 nM T66383 CAJ4V9 8359 IC50 = 2900 nM T66383 CJ49WT 3784000 Ki = 500000 nM T66383 CGP65C 10003390 IC50 = 3700 nM T66383 CJX25F 45267877 Ki = 500000 nM T66383 C0U7QJ 57520253 IC50 = 3 nM T66383 CPDT85 57520354 IC50 = 30000 nM T66383 C2N3RA 57520356 IC50 = 45 nM T66383 CL5W3O 68283281 IC50 = 2 nM T66383 CV0IW5 68283802 IC50 = 700 nM T66383 C17JAZ 68284084 IC50 = 500 nM T66383 CD3P0Z 68284292 IC50 = 450 nM T66383 CD19EU 68284568 IC50 = 22000 nM T66383 C6QNX1 68284579 IC50 = 650 nM T66383 CW70TJ 68284602 IC50 = 50 nM T66383 CYCN51 68284666 IC50 = 1400 nM T66383 CW21KG 68284716 IC50 = 500 nM T66383 CN83VA 68284837 IC50 = 850 nM T66383 CC5X2I 71009356 IC50 = 24750 nM T66383 CLZ3Q2 71009390 IC50 = 10 nM T66383 CK0BD4 71009508 IC50 = 12 nM T66383 C57XVO 71009528 IC50 = 150 nM T66383 C3C4YV 71009592 IC50 = 320 nM T66383 C1DUO9 71009649 IC50 = 50 nM T66383 CGF63Y 71009743 IC50 = 30 nM T66383 C8YV5A 71042234 IC50 = 300 nM T66383 CRL5H0 72705807 IC50 = 2 nM T66383 CJP25I 72720766 IC50 = 3 nM T66383 CF7Y9K 72720769 IC50 = 6 nM T66383 CMG39E 86673884 IC50 = 11 nM T66383 CJT6F2 89184242 IC50 = 66 nM T66383 C4VL5T 90480060 IC50 = 13600 nM T66383 CQG9T0 90480064 IC50 = 120 nM T66383 CC1QY8 91758756 IC50 = 100 nM T66383 CKZ75W 117819609 IC50 = 270 nM T66383 CL8WC6 117819668 IC50 = 260 nM T66383 CNY29S 117819734 IC50 = 8 nM T66383 CYR7U4 117819978 IC50 = 2500 nM T66383 C2W5BU 117820065 IC50 = 3 nM T66383 CEI6Y5 117820116 IC50 = 15 nM T66383 CG6S9U 117820135 IC50 = 30 nM T66383 C5R7OY 117820157 IC50 = 20 nM T66383 CI4ZR0 117820213 IC50 = 25 nM T66383 C2RXZ3 117820231 IC50 = 8 nM T66383 CI5EW6 117820295 IC50 = 5 nM T66383 C4HAT8 117820303 IC50 = 10 nM T66383 C3WOY4 118074135 IC50 = 100 nM T66383 CO9P5Y 118207089 IC50 = 22 nM T66383 CW8SX7 118796776 IC50 = 6 nM T66383 C1JSV9 121379599 IC50 = 23 nM T66383 CKJN32 122164799 IC50 = 14000 nM T66383 CGY9X5 122164804 IC50 = 5800 nM T66383 CP5K0Z 122177127 IC50 = 27.31 nM T66383 CM47NU 122177128 IC50 = 77 nM T66383 C7WPT8 130301786 IC50 = 23 nM T66383 CPWD42 130301808 IC50 = 150 nM T66383 COM3F6 132471826 IC50 = 20000 nM T66383 CO9H4P 134145794 IC50 = 31.95 nM T66383 CEN98J 134147033 IC50 = 19 nM T66383 C3D1WS 134158401 IC50 = 20000 nM T66383 CWDG03 134158402 IC50 = 75000 nM T66383 COTM78 134158403 IC50 = 84000 nM T66383 C8QX6N 134158404 IC50 = 120000 nM T66383 CK74OV 134158405 IC50 = 32000 nM T66383 CSXH80 137632616 IC50 > 30000 nM T66383 CUBF84 137647883 IC50 = 15 nM T66383 CF50JP 137652109 IC50 = 370 nM T66383 CLJ2T7 137654246 IC50 = 17000 nM T66383 C8XO2B 145950935 IC50 = 3400 nM T66383 C5IFD0 145951043 IC50 = 44000 nM T66383 CX91NP 145953441 IC50 = 43000 nM T66383 CWM3I0 145953577 IC50 = 310000 nM T66383 CP5S6G 145959105 IC50 = 257000 nM T66383 CR39WC 145959425 IC50 = 98000 nM T66383 C5WUD2 145971969 IC50 = 690000 nM T66383 CP91BA 145972685 IC50 = 140000 nM T66383 C5X4VB 155520208 IC50 = 8200 nM T66383 CM5LO9 155552558 IC50 = 64000 nM T66383 D04MIN 57412074 IC50 = 1 nM T47657 D0AF6O 71731823 IC50 = 2.7 nM T47657 D0E3TC 44259 IC50 = 3.6 nM T47657 D0Y2PO 71770709 IC50 = 10600 nM T47657 C5VPH9 16129448 IC50 = 360 nM T47657 CYT37A 46232443 IC50 > 50000 nM T47657 C48ZVW 46232555 IC50 = 18000 nM T47657 CS9B1U 46232556 IC50 = 10000 nM T47657 CPHX64 57325478 IC50 > 50000 nM T47657 CQ9BW4 57325479 IC50 > 50000 nM T47657 CVK0G4 58056356 IC50 > 50000 nM T47657 C37NKO 67129970 IC50 = 7400 nM T47657 CK80LJ 67130050 IC50 = 6010 nM T47657 CV63UL 67240318 IC50 > 10000 nM T47657 C7GRV2 68755406 IC50 > 10000 nM T47657 CPG3A5 86302574 IC50 > 30000 nM T47657 CKS28E 127034802 IC50 = 43.1 nM T47657 CUO0C5 132156633 IC50 > 10000 nM T47657 C25ERN 137631967 IC50 = 45.3 nM T47657 CI1E8V 137634241 IC50 = 5110 nM T47657 C06JRX 137637094 IC50 = 122.9 nM T47657 C1DK0P 137651391 IC50 = 68.5 nM T47657 CV5H3Z 137657932 IC50 = 299.5 nM T47657 CZ9BN4 138320062 IC50 = 0.567 nM T47657 C2MD1Q 155513187 IC50 > 10000 nM T47657 C78MZC 155536330 IC50 = 4 nM T47657 D0K5UF 72710568 IC50 = 2 nM T51102 D0E3TC 44259 IC50 < 100 nM T51102 CGAN35 2856 IC50 = 16000 nM T51102 C18WEB 490561 IC50 < 100 nM T51102 CYZU17 937050 IC50 = 13000 nM T51102 CLG63C 1530863 IC50 = 9400 nM T51102 CZ5KB1 2455709 IC50 = 12000 nM T51102 CVB83T 5330811 IC50 = 8000 nM T51102 C2NP5X 6897738 IC50 = 11000 nM T51102 C2WG8I 7216437 IC50 = 11000 nM T51102 C7L3JN 9124464 IC50 = 13000 nM T51102 C5B3XJ 11620410 IC50 > 40000 nM T51102 CV56YS 16414650 IC50 = 20000 nM T51102 CQOT74 16805560 IC50 = 15000 nM T51102 CJCQ86 17395684 IC50 = 19000 nM T51102 C6QT0J 44622837 IC50 > 1000 nM T51102 CU9GM5 53307873 Ki = 3400 nM T51102 CXB94H 53466728 IC50 > 10000 nM T51102 CYQ41S 53466951 IC50 = 978 nM T51102 CX0R1K 53469059 IC50 = 905 nM T51102 CV7C0D 53469060 IC50 = 359 nM T51102 CCKD45 53469061 IC50 = 99 nM T51102 C91STB 53469449 IC50 = 291 nM T51102 CZ1CI3 53469824 IC50 > 10000 nM T51102 CQEA01 56659460 IC50 > 100000 nM T51102 C5KEW0 56659461 IC50 = 3000 nM T51102 C7PCY5 56659462 IC50 > 100000 nM T51102 C1JD8Z 56659512 IC50 = 12000 nM T51102 C34VCR 56659514 IC50 = 90000 nM T51102 CPQ2A9 56659515 IC50 = 9000 nM T51102 CYK40N 56659516 IC50 > 100000 nM T51102 C39BXF 56659517 IC50 = 600 nM T51102 CD65YZ 56662919 IC50 = 1500 nM T51102 C6MR1L 56662961 IC50 = 1500 nM T51102 C8XKC2 56662962 IC50 > 100000 nM T51102 C0T8QZ 56662963 IC50 = 100 nM T51102 COH9G3 56666393 IC50 = 48000 nM T51102 CJD0P8 56666438 IC50 > 100000 nM T51102 C36XYF 56666439 IC50 = 18000 nM T51102 CA42FJ 56666467 IC50 = 11000 nM T51102 C3JT6B 56669804 IC50 = 300 nM T51102 C6X5UV 56669805 IC50 = 8000 nM T51102 C1Q8AD 56669806 IC50 = 100 nM T51102 CG1IT9 56669852 IC50 = 1500 nM T51102 CND1T2 56669853 IC50 = 50000 nM T51102 CM5FL6 56673297 IC50 = 55000 nM T51102 CA32UJ 56673389 IC50 = 14000 nM T51102 C87RUH 56673390 IC50 = 12000 nM T51102 CET8S0 56676623 IC50 = 19000 nM T51102 CM40ON 56676624 IC50 = 51000 nM T51102 CHR3M8 56676675 IC50 > 100000 nM T51102 C30BIC 56676676 IC50 = 45000 nM T51102 CEZ39Y 56679958 IC50 = 3500 nM T51102 CW04DN 56679959 IC50 = 2500 nM T51102 CDEM30 56679960 IC50 = 7000 nM T51102 CB1H6Z 56679961 IC50 > 100000 nM T51102 CH1UK6 56680023 IC50 = 750 nM T51102 C5KB4E 56680024 IC50 = 11000 nM T51102 CS1U2A 56683286 IC50 > 100000 nM T51102 CGX39M 56683287 IC50 = 150 nM T51102 CUO35I 56683288 IC50 = 50000 nM T51102 CKF34Z 56683289 IC50 > 100000 nM T51102 C3P0FG 56683334 IC50 > 100000 nM T51102 CX4H6I 86583042 IC50 > 10000 nM T51102 C4TXF2 118730409 IC50 = 480000 nM T51102 CW3OF5 135398511 IC50 < 100 nM T51102 C5L7IE 135411750 IC50 = 10500 nM T51102 C5RNG3 135432788 IC50 = 4000 nM T51102 C2D5WG 135653128 IC50 = 3000 nM T51102 CXC69T 137321158 IC50 = 210 nM T51102 C2MD1Q 155513187 IC50 > 10000 nM T51102 D02PVB 8515 IC50 = 8000 nM T51102 D04WFN 10202471 IC50 = 2000 nM T51102 D06KDU 16760346 IC50 = 7000 nM T51102 D06KSF 9549300 IC50 = 250 nM T51102 D07OCA 5330812 IC50 = 1600 nM T51102 D09RES 11665831 IC50 = 12000 nM T51102 D0A7FQ 11644425 IC50 = 5000 nM T51102 D0D2FC 2794188 IC50 = 3000 nM T51102 D0D5HQ 5330797 IC50 = 6000 nM T51102 D0E0XV 9903786 IC50 = 250 nM T51102 D0HZ8U 3467590 IC50 < 100 nM T51102 D0L3FK 5289419 IC50 = 5000 nM T51102 D0N4LR 53469448 IC50 = 696 nM T51102 D0Q3EW 9549303 IC50 = 20000 nM T51102 D0Q7TO 6419766 IC50 = 15000 nM T51102 D0R5FH 438981 IC50 = 6000 nM T51102 D0T8KR 9549289 IC50 = 4000 nM T51102 D0Y0BK 11524144 IC50 = 16000 nM T51102 D0Y0ES 3707 IC50 < 100 nM T51102 D0Z2CN 135418335 IC50 < 100 nM T56051 D03GET 4055 IC50 = 290000 nM T56051 CZ9A4Y 756803 Ki = 1200 nM T56051 C1PC4Y 756804 Ki = 910 nM T56051 CZ2TO3 1948620 Ki > 30000 nM T56051 CS9RO8 2729042 IC50 = 75000 nM T56051 C4DQ7P 11222830 IC50 = 3000 nM T56051 CXL01A 16760696 Ki = 400 nM T56051 CC0V1O 23628286 Ki = 740 nM T56051 CC21QM 44440958 Ki > 30000 nM T56051 CT74NW 44440961 Ki = 10000 nM T56051 CH36OC 44440963 Ki = 1400 nM T56051 CSA2Y9 44440965 Ki = 30000 nM T56051 C0B2YS 44440967 Ki = 5300 nM T56051 C7AL0R 44440969 Ki = 3600 nM T56051 CB9O2D 44440971 Ki = 30000 nM T56051 C5XZH6 44440974 Ki = 11000 nM T56051 CGVU60 44440976 Ki = 1500 nM T56051 CC9K6Q 44440979 Ki = 30000 nM T56051 CL3U8X 44440981 Ki = 20000 nM T56051 C67WDH 44440983 Ki > 30000 nM T56051 CFE63C 44440985 Ki = 20000 nM T56051 C74IUM 44440987 Ki = 2000 nM T56051 CNW72F 44440990 Ki > 30000 nM T56051 CG12PE 45265922 Ki = 2800 nM T56051 C3Z5CV 46830074 IC50 > 200000 nM T56051 C3P8EW 52940990 IC50 = 940 nM T56051 CEW74T 52942184 IC50 = 126000 nM T56051 CU0H7T 52943029 IC50 = 810 nM T56051 CA6BT2 52944213 IC50 = 880 nM T56051 D0N6BC 950368 Ki = 2300 nM T56051 D0Y7OI 11563133 IC50 = 22300 nM T51408 D04KJO 3410 EC50 = 25.12 nM T51408 D04PHC 5816 EC50 = 31 nM T51408 D07MOX 439260 EC50 = 5.5 nM T51408 D0CQ0Z 33630 Ki = 515 nM T51408 D0G8NN 119570 Ki > 10000 nM T51408 D0I8FI 3779 EC50 = 0.97 nM T51408 D0L5YV 5152 EC50 = 1000 nM T51408 D07NFW 9870286 Ki = 21 nM T51408 D07WHS 5312115 EC50 = 220 nM T51408 D0A5EF 9887812 EC50 = 3.981 nM T51408 D0DH5X 44472635 EC50 = 1.1 nM T51408 D0I2XM 3038500 EC50 = 2 nM T51408 D0LI1C 44469321 IC50 > 30000 nM T51408 D0MT5C 16118894 EC50 = 1.6 nM T51408 D01SWK 5493324 EC50 = 0.016 nM T51408 D02KMG 9892481 EC50 = 39.81 nM T51408 D03GLM 9828292 Ki = 9 nM T51408 D04YJU 9829836 EC50 = 0.43 nM T51408 D0Y1PG 9841972 EC50 = 0.095 nM T51408 CYG2P9 2755 EC50 = 10000 nM T51408 CJQE97 5581 EC50 = 1.7 nM T51408 C5H9CN 9287 Ki > 10000 nM T51408 CXS0V8 26162 Ki = 4100 nM T51408 C96ASF 164451 Ki = 520 nM T51408 C9G0KB 213051 EC50 = 1.2 nM T51408 CPA9F2 443372 EC50 = 39.81 nM T51408 C17WFV 2770390 Ki = 3100 nM T51408 CRS35B 2796082 EC50 = 120 nM T51408 CD19NG 3654892 Ki > 10000 nM T51408 CMSB89 3687256 Ki = 411 nM T51408 C1CK2S 4143663 Ki = 1180 nM T51408 CBC7N9 4276762 Ki = 3380 nM T51408 CW2IR6 4421983 Ki = 409 nM T51408 C70GLP 5187268 Ki = 1480 nM T51408 C1MW2P 6916441 EC50 = 0.062 nM T51408 C7SIU5 9799092 EC50 = 15.85 nM T51408 CH6PX1 9801145 EC50 = 7.943 nM T51408 C7ZQ3D 9803765 EC50 = 220 nM T51408 C68VZH 9803988 EC50 = 16 nM T51408 CRJ79X 9804536 EC50 = 2.086 nM T51408 CUY3S0 9810596 EC50 = 19 nM T51408 C7W1VG 9820697 EC50 = 300 nM T51408 CM48YW 9821129 EC50 = 630 nM T51408 CD7TA2 9823696 EC50 = 1.585 nM T51408 CD2U3O 9826638 EC50 = 13 nM T51408 CY8U3K 9826916 EC50 = 30 nM T51408 CB6O2M 9827999 EC50 = 20 nM T51408 CSZY30 9828477 EC50 = 6 nM T51408 CYR8O6 9831168 EC50 = 66 nM T51408 CK7WI5 9832011 EC50 = 16 nM T51408 C30LWX 9837752 Ki = 17000 nM T51408 CK7DS2 9842600 EC50 = 39 nM T51408 C3JYI0 9845280 EC50 = 158.49 nM T51408 C1CEO4 9845282 EC50 = 0.1 nM T51408 C0OS8W 9847067 EC50 = 25.12 nM T51408 CY3DL8 9849126 EC50 = 199.53 nM T51408 C9FAP3 9853471 EC50 = 6 nM T51408 CB6R3T 9858463 EC50 = 20 nM T51408 CR7X5O 9858464 EC50 = 200 nM T51408 CJIR63 9871386 EC50 = 12.59 nM T51408 CJ72CL 9871525 EC50 = 59 nM T51408 C1L6XP 9871887 Ki = 21.38 nM T51408 CL54GH 9872113 Ki = 160 nM T51408 C51FVW 9872550 EC50 = 2.4 nM T51408 CVF5O3 9873245 EC50 = 49 nM T51408 CSRF54 9873257 EC50 = 13 nM T51408 CDQ84R 9888047 EC50 = 0.2512 nM T51408 C5L3VF 9893058 EC50 = 50.12 nM T51408 CVR17A 9895810 Ki = 93 nM T51408 CRV61G 9896742 EC50 = 78 nM T51408 CMC06V 9896817 EC50 = 140 nM T51408 CFI97S 9904205 IC50 = 1862.09 nM T51408 CYWQ50 9906447 Ki > 10000 nM T51408 CQP6X3 9906822 EC50 = 0.36 nM T51408 CQ27DF 9907863 EC50 = 489.78 nM T51408 CUHF02 9908924 EC50 = 60 nM T51408 C2A1CZ 9912443 EC50 = 6 nM T51408 CMH72E 9912580 EC50 = 5.9 nM T51408 CDH69A 9915235 EC50 = 20 nM T51408 CYH07G 9915238 EC50 = 6.3 nM T51408 CR1T5X 9915920 EC50 = 120 nM T51408 CH9OT6 9917962 EC50 = 13 nM T51408 CW7YJ1 9924779 EC50 = 42 nM T51408 C1XSL4 9927453 EC50 = 0.36 nM T51408 C92XMC 9933039 EC50 = 6.3 nM T51408 C7MO0Z 9938030 EC50 = 12 nM T51408 CZM1E2 9946573 EC50 = 57 nM T51408 C92NVH 9947212 EC50 = 265 nM T51408 C9PVT1 9947512 EC50 = 170 nM T51408 CM13QP 9957065 Ki = 33 nM T51408 CCN27K 9958539 EC50 = 800 nM T51408 CM6I4O 9960584 Ki = 6 nM T51408 CCA49K 9962058 EC50 = 600 nM T51408 CB3AQ9 9967732 EC50 = 37 nM T51408 CFTV18 9984028 EC50 = 6.31 nM T51408 C1NYC0 10002049 EC50 = 0.6 nM T51408 CEF4Y3 10003858 EC50 = 0.14 nM T51408 CO3DB4 10007337 EC50 = 23 nM T51408 CP0H1B 10008017 EC50 = 8 nM T51408 CTE2I9 10048077 EC50 = 4.8 nM T51408 CWJ25B 10054165 EC50 = 5.7 nM T51408 CRU28L 10054896 EC50 = 8 nM T51408 CBVG28 10075383 EC50 = 0.77 nM T51408 CVE2T1 10076176 EC50 = 794.33 nM T51408 C8TBK0 10076548 EC50 = 9 nM T51408 C7SL6M 10076885 EC50 = 13 nM T51408 CP7WF3 10092953 EC50 = 1.8 nM T51408 CSNP15 10099346 EC50 = 14 nM T51408 CL81PN 10099459 EC50 = 18 nM T51408 CRK6B0 10101116 EC50 = 57 nM T51408 C54EYD 10108561 IC50 < 1000 nM T51408 CP6L3C 10112732 EC50 = 100 nM T51408 CA4MV1 10112744 EC50 = 65 nM T51408 C73TAD 10112753 EC50 = 36 nM T51408 C8SAN2 10113837 EC50 = 0.5 nM T51408 CQW48U 10117815 Ki = 25 nM T51408 CE90NU 10118962 EC50 = 18 nM T51408 CJ31XM 10119061 EC50 = 100 nM T51408 C6G4BM 10119452 Ki = 24 nM T51408 CLB01Q 10119515 EC50 = 37 nM T51408 C07WRX 10121328 EC50 = 43 nM T51408 CZJB20 10121514 EC50 = 10 nM T51408 CIX83H 10131985 EC50 = 309 nM T51408 CCRO89 10132882 EC50 = 170 nM T51408 CE27RV 10135864 EC50 = 21 nM T51408 CZ8AQ7 10136220 EC50 = 290 nM T51408 C0G7FS 10138551 EC50 = 25 nM T51408 C8ZK3L 10138809 EC50 = 42 nM T51408 CZ0J7I 10140092 Ki = 53 nM T51408 CP0K9U 10140428 EC50 = 120 nM T51408 CTZ03I 10140889 EC50 = 36 nM T51408 C4B7XL 10140996 Ki = 8 nM T51408 C0FS3J 10142284 EC50 = 80 nM T51408 C1UKY7 10143516 EC50 > 2000 nM T51408 CO3F6S 10144004 EC50 = 850 nM T51408 CD0RL9 10145446 EC50 = 20 nM T51408 CHZQ30 10145482 EC50 = 29 nM T51408 CDHS42 10155942 EC50 = 47 nM T51408 CCP74I 10160281 EC50 = 665 nM T51408 C27MZY 10160636 EC50 = 150 nM T51408 C7YM0K 10160869 EC50 = 10 nM T51408 CGJ10H 10162297 Ki = 110 nM T51408 C02SXI 10162876 EC50 = 23 nM T51408 C7URQ6 10166311 EC50 = 26 nM T51408 C39HYQ 10168241 EC50 = 200 nM T51408 C2B5SJ 10180440 EC50 = 40 nM T51408 CGN3F7 10182229 EC50 = 41 nM T51408 C7AOJ4 10182494 EC50 = 464 nM T51408 C6P8SU 10183066 EC50 = 4 nM T51408 CEAM37 10183401 EC50 = 537 nM T51408 C50VQT 10186687 EC50 = 1020 nM T51408 C0YJ2G 10186965 Ki = 7 nM T51408 CB9HW6 10187201 EC50 = 8 nM T51408 C8EOD0 10187653 EC50 = 135 nM T51408 CBT5M6 10188669 EC50 = 36 nM T51408 CZHJ01 10189730 EC50 = 1 nM T51408 CEXA73 10193354 EC50 = 520 nM T51408 CU01VL 10200545 EC50 = 38 nM T51408 C1H8AB 10201549 EC50 = 200 nM T51408 CCO4D7 10202842 EC50 = 30 nM T51408 C56USA 10203169 EC50 = 31.62 nM T51408 CM2I8S 10203259 EC50 = 1360 nM T51408 CL1UB7 10204992 EC50 = 8 nM T51408 C6Y5JB 10205362 EC50 = 89 nM T51408 C9N1WB 10205463 EC50 = 90 nM T51408 CF5RL8 10206782 EC50 = 26 nM T51408 C2MX7I 10207208 Ki = 9 nM T51408 C1H0JA 10207209 Ki = 150 nM T51408 CV0DC6 10209114 EC50 = 290 nM T51408 C3A2UK 10209243 EC50 = 10.6 nM T51408 C2KEW4 10209574 EC50 = 23 nM T51408 CD59TX 10211392 EC50 = 55 nM T51408 CF6R2U 10217757 EC50 = 3.162 nM T51408 C70MAV 10222907 EC50 = 99 nM T51408 CL1MU9 10225274 EC50 = 7 nM T51408 CPE8M6 10225563 EC50 = 5.012 nM T51408 C2I6BY 10227108 Ki = 460 nM T51408 CR2TZ8 10230413 Ki = 6 nM T51408 CG93UN 10230721 EC50 = 380 nM T51408 C3A0ZR 10230922 EC50 > 2000 nM T51408 C4KTP1 10231394 EC50 = 58 nM T51408 C9Y4AT 10231679 Ki = 19 nM T51408 CF4Z1B 10232096 EC50 = 250 nM T51408 CV4QB7 10232593 EC50 = 66 nM T51408 C2YDG7 10233153 EC50 = 9 nM T51408 CSC3V2 10238776 EC50 = 7.943 nM T51408 CDCP62 10239722 EC50 = 10 nM T51408 CYBX59 10258518 EC50 = 0.93 nM T51408 CE36WH 10271144 EC50 = 943 nM T51408 C1KR8D 10273469 EC50 = 580 nM T51408 CL81ST 10273529 EC50 = 1460 nM T51408 C8HIN2 10273799 EC50 = 165 nM T51408 CBW0X8 10274448 EC50 = 180 nM T51408 CBFQ89 10275157 EC50 = 47 nM T51408 CV25SE 10278987 EC50 = 90 nM T51408 C01JVZ 10280222 EC50 = 126 nM T51408 C1EZ4U 10280301 EC50 = 41 nM T51408 C6YUK7 10281165 EC50 = 60 nM T51408 C9TLW7 10282871 EC50 = 11 nM T51408 CO24KP 10283146 EC50 = 11 nM T51408 CF4Y7P 10283539 EC50 = 1 nM T51408 C5TEI1 10288976 EC50 = 39.81 nM T51408 C7F6LZ 10291064 EC50 = 27 nM T51408 CD1S6J 10292413 EC50 = 57 nM T51408 C0Z6CM 10294264 EC50 = 299 nM T51408 C2SFK0 10295131 EC50 = 9900 nM T51408 C6QBA8 10296491 EC50 = 24 nM T51408 C2J7WF 10296855 EC50 = 617 nM T51408 CV42BX 10297331 EC50 = 220 nM T51408 CIW29S 10298567 EC50 = 0.8 nM T51408 CS21VJ 10301056 EC50 = 47 nM T51408 C2FSP4 10301101 EC50 = 60 nM T51408 C3RP8X 10301445 EC50 = 70 nM T51408 CUJ3M7 10302342 EC50 = 50 nM T51408 C1U3DW 10302915 EC50 = 32 nM T51408 C9PK4A 10304565 EC50 = 45 nM T51408 COES23 10304786 EC50 = 48 nM T51408 CUML26 10305108 EC50 = 5 nM T51408 C1PSZ4 10346448 EC50 = 1.259 nM T51408 CZ26AE 10347866 EC50 = 14 nM T51408 C7H9PZ 10371216 EC50 = 6 nM T51408 CDAC63 10381889 IC50 = 870.96 nM T51408 CDRL02 10393774 EC50 = 4 nM T51408 C5QI3T 10416448 EC50 = 3.1 nM T51408 C6URQ9 10416656 EC50 = 13 nM T51408 C6ZIY2 10437614 EC50 = 3.6 nM T51408 C59OLP 10438390 EC50 = 7.2 nM T51408 CA20IB 10483845 EC50 = 14 nM T51408 CQKI17 10544781 Ki = 67608.3 nM T51408 CQ4Z8H 10553602 EC50 = 60 nM T51408 CL0MJ3 10553603 EC50 = 130 nM T51408 CK87QN 10575455 EC50 = 20 nM T51408 CB83SX 10601234 EC50 = 66 nM T51408 C4NWL1 10602703 EC50 = 26 nM T51408 CW2S8I 10626150 EC50 = 15 nM T51408 C28DCI 10627031 EC50 = 92 nM T51408 CWP9M1 10627736 EC50 = 6.9 nM T51408 C51DIX 10648298 EC50 = 39 nM T51408 CX9WA0 10651078 EC50 = 7.6 nM T51408 C1C6KV 10651147 EC50 = 4 nM T51408 CS4FX5 10697841 EC50 = 98 nM T51408 CXPN86 10718924 EC50 = 270 nM T51408 C8WX4M 10722793 EC50 = 4.3 nM T51408 C6R5QN 10745501 EC50 = 36 nM T51408 CFJA38 10746499 EC50 = 53 nM T51408 CQA4E2 10841171 EC50 = 19 nM T51408 CHM6J4 10841426 EC50 = 6.3 nM T51408 C05CGB 10863093 EC50 = 5.012 nM T51408 C92OSW 10902809 EC50 = 19.95 nM T51408 CSF82D 10915880 EC50 = 5754.4 nM T51408 CY1QM6 10940242 EC50 = 10 nM T51408 C3OFL7 10981769 EC50 = 610 nM T51408 CC6V1Z 11002571 EC50 = 794.33 nM T51408 CRJ5L3 11003341 EC50 = 25.12 nM T51408 C8V7XF 11005613 EC50 = 19.95 nM T51408 C6TAO1 11026016 EC50 = 19.95 nM T51408 CCKZ08 11038599 EC50 = 15.85 nM T51408 CZI9B1 11060184 EC50 = 0.7943 nM T51408 C23NHX 11091850 EC50 = 63.1 nM T51408 C2N0BD 11124502 EC50 = 1.585 nM T51408 C8FVK0 11134054 EC50 = 1.259 nM T51408 C41RIK 11152564 EC50 = 6.5 nM T51408 C62GDB 11156916 EC50 = 0.1259 nM T51408 C5N7WZ 11163954 EC50 = 69 nM T51408 C8Y9VL 11165102 EC50 = 2.8 nM T51408 C34JRO 11169365 EC50 = 63.1 nM T51408 CY04IB 11180293 EC50 = 39.81 nM T51408 CZL0Y7 11187476 EC50 = 1.7 nM T51408 CY46ON 11189002 EC50 = 38 nM T51408 CG3DV6 11199616 EC50 = 0.96 nM T51408 CNJ7I5 11221586 EC50 = 12 nM T51408 CI5LY3 11221652 EC50 = 1.7 nM T51408 C10HWX 11222097 EC50 = 22 nM T51408 CUGE45 11224220 EC50 = 0.14 nM T51408 CB69KG 11224275 EC50 = 0.43 nM T51408 CX6EI1 11235459 EC50 = 0.26 nM T51408 CZU17C 11236495 EC50 = 70 nM T51408 CUSR07 11244811 EC50 = 96 nM T51408 CD2VF8 11268355 EC50 = 0.15 nM T51408 CNJZ06 11270069 EC50 = 13 nM T51408 CBJ49T 11270071 EC50 = 11 nM T51408 CRFS12 11272641 EC50 = 0.13 nM T51408 CJ4CE6 11324939 EC50 = 0.97 nM T51408 CQ08YH 11340895 EC50 = 0.46 nM T51408 CGQ2D0 11342656 EC50 = 12 nM T51408 CAV5Q7 11349698 EC50 = 14 nM T51408 CUNJ91 11352782 EC50 = 0.32 nM T51408 CPCN92 11360474 EC50 = 28 nM T51408 CH3UO2 11373418 EC50 = 0.92 nM T51408 C0MG9U 11381882 EC50 = 33 nM T51408 C0YB8T 11398536 EC50 = 0.14 nM T51408 CYWD16 11419142 EC50 = 11 nM T51408 CMX29E 11420551 EC50 = 0.6 nM T51408 CQC36P 11432806 EC50 = 0.21 nM T51408 CL1M5W 11453340 EC50 = 0.56 nM T51408 C6TA1B 11476004 EC50 = 0.81 nM T51408 CW3YR2 11495581 EC50 = 31.62 nM T51408 CZ62AI 11546349 EC50 = 31.62 nM T51408 CAWR47 11556330 EC50 = 5 nM T51408 CWM5K6 11575154 EC50 = 0.1 nM T51408 CP2WJ8 11592062 EC50 = 25.12 nM T51408 CY15EM 11605652 EC50 = 19952.62 nM T51408 CA0R9K 11611195 EC50 = 7.4 nM T51408 C7ZTC8 11647543 EC50 = 0.2512 nM T51408 C1J4XV 11661536 EC50 = 63.1 nM T51408 COHD32 11669967 EC50 = 0.1995 nM T51408 CD31TA 11718543 EC50 = 39.81 nM T51408 CT1OL3 11758172 EC50 = 7.1 nM T51408 C2UN8W 11785699 EC50 = 1 nM T51408 C4ISZ7 11810896 EC50 = 12.59 nM T51408 C13CET 11810992 EC50 = 3.8 nM T51408 C8JQL7 11957735 IC50 > 10000 nM T51408 C3BXJ2 12017001 EC50 = 39 nM T51408 CF5TK1 12017002 EC50 = 37 nM T51408 C38DZJ 12017003 EC50 = 35 nM T51408 CN5A2D 12017004 EC50 = 11 nM T51408 C40KFM 12017005 EC50 = 15 nM T51408 C0G3XR 12017006 EC50 = 22 nM T51408 C2FZ3H 12017007 EC50 = 35 nM T51408 CDZQ57 12017010 EC50 = 5.2 nM T51408 CEC98K 12017011 EC50 = 4 nM T51408 C02SVL 12017012 EC50 = 4.3 nM T51408 C1ZH0K 12017013 EC50 = 19 nM T51408 C31JDV 12017014 EC50 = 9.2 nM T51408 CLIX97 12017015 EC50 = 19 nM T51408 CO0ST4 12017016 EC50 = 5.3 nM T51408 C7Z8WC 12017017 EC50 = 2.3 nM T51408 C60OVP 12017018 EC50 = 210 nM T51408 CPU75A 12043155 EC50 = 29 nM T51408 C1MFE0 12043156 EC50 = 15 nM T51408 CR0T9I 12043157 EC50 = 19 nM T51408 C4U9KY 12043158 EC50 > 100 nM T51408 CW0XL2 12043159 EC50 = 130 nM T51408 CK4ZC5 12047933 Ki = 17000 nM T51408 C7I2CM 12049914 EC50 = 52 nM T51408 C5M8FQ 12049915 EC50 = 24 nM T51408 C49XHR 12049916 EC50 = 14 nM T51408 C7TAQ6 12049917 EC50 = 22 nM T51408 CDI75Z 12049918 EC50 = 18 nM T51408 C0LF7J 12049919 EC50 = 6.4 nM T51408 C6JWS8 12049920 EC50 = 14 nM T51408 CU7A5R 12049921 EC50 = 24 nM T51408 CDZF95 12049922 EC50 = 4.1 nM T51408 CZ4V2K 12049923 EC50 = 48 nM T51408 C8DUY7 12049924 EC50 = 10 nM T51408 CF0IG7 12049925 EC50 = 11 nM T51408 C3U1SP 12049926 EC50 = 14 nM T51408 C91IBR 12114484 EC50 = 70 nM T51408 C6KUG7 12147062 EC50 = 9 nM T51408 CFC0D6 14823035 EC50 = 420 nM T51408 CKFL78 15221053 EC50 = 2760 nM T51408 C9HLK1 15221055 EC50 = 27595 nM T51408 C25CVZ 15483879 EC50 = 18 nM T51408 CLNE19 15483880 EC50 = 12 nM T51408 CUK85J 15483883 EC50 = 8 nM T51408 CSDO83 15523859 EC50 = 2.2 nM T51408 C6Q9FZ 15523860 EC50 = 5.9 nM T51408 CKP61A 15523861 EC50 = 4.2 nM T51408 CH8KY4 16126657 EC50 = 10.1 nM T51408 C42ELY 16219010 EC50 = 25.12 nM T51408 CDV38P 16222840 EC50 = 0.35 nM T51408 C9ONT1 16222940 EC50 = 0.066 nM T51408 C3C9WR 16223045 EC50 = 0.23 nM T51408 CHJ65G 16223251 EC50 = 0.059 nM T51408 CZ2IS9 16660294 Ki > 10000 nM T51408 CH2M3I 18435422 Ki = 7300 nM T51408 CL2I9W 18435434 Ki = 1100 nM T51408 C09BQZ 18662692 Ki = 70 nM T51408 C4BK1Y 18662693 Ki = 74 nM T51408 C4WY2J 18662695 Ki = 8600 nM T51408 C5PU4B 18662696 Ki = 120 nM T51408 CLO48S 18662698 Ki = 800 nM T51408 C0X6JR 18662700 Ki = 30000 nM T51408 CIH6K0 18662704 Ki = 8 nM T51408 CJ20DY 18662710 Ki = 33000 nM T51408 C97NET 18662711 Ki = 77 nM T51408 C0T4FJ 18662712 Ki = 3100 nM T51408 CS4VL7 18662714 Ki = 9600 nM T51408 C79GPY 18662716 Ki = 33 nM T51408 CH0JA9 18662718 Ki = 89 nM T51408 CPZX38 18662719 Ki = 8.8 nM T51408 CU96BJ 18662720 Ki = 10000 nM T51408 C1TA5E 18662723 Ki = 7000 nM T51408 CG7L2C 19073112 Ki = 87000 nM T51408 C4E6TA 19073116 Ki = 414 nM T51408 C48KSO 19073121 Ki = 129 nM T51408 C4P5KH 19073136 Ki = 70 nM T51408 CI51VS 19073138 Ki = 44 nM T51408 CN5GI8 19073142 Ki = 520 nM T51408 C52MPD 19073145 Ki = 440 nM T51408 C8W5XC 19073158 Ki = 360 nM T51408 CG6R2K 19073196 Ki = 133 nM T51408 CPN98A 19073202 Ki = 1600 nM T51408 CQF4J3 19073210 Ki = 480 nM T51408 C45RWV 19073229 Ki = 700 nM T51408 C2L0HA 19073276 Ki = 230 nM T51408 CWJ7K6 19360455 EC50 = 200 nM T51408 C9JD5Y 19360456 EC50 = 20 nM T51408 C3T5HF 21509921 Ki > 10000 nM T51408 C72IMX 22171479 EC50 > 100 nM T51408 C7PQ8B 22171507 EC50 = 12 nM T51408 CCMB98 22171637 EC50 = 48 nM T51408 CN9Z2S 23661589 EC50 = 0.0631 nM T51408 CWEM23 24321330 Ki = 1030 nM T51408 CR2HF1 24812040 EC50 = 4.9 nM T51408 CE5B9G 24812041 EC50 = 3.9 nM T51408 C0F7KH 24812042 EC50 = 3.4 nM T51408 CHA4O9 24812043 EC50 = 181 nM T51408 C4Q3XY 24812044 EC50 = 2.7 nM T51408 CH3UP8 24812045 EC50 = 235 nM T51408 CM78DS 24812046 EC50 = 136 nM T51408 CA3MI7 24812154 EC50 = 3.8 nM T51408 CRV58X 24822304 EC50 = 8.7 nM T51408 CST3O6 24822310 EC50 = 6.7 nM T51408 C3C7SF 24822313 EC50 = 91 nM T51408 CTJD72 24822469 EC50 = 7.5 nM T51408 CIWN92 24822472 EC50 = 15 nM T51408 C8F7MR 24822643 EC50 = 4.9 nM T51408 C86IOK 24822645 EC50 = 2 nM T51408 CN4H3E 24822648 EC50 = 0.62 nM T51408 C4H6MR 24822815 EC50 = 0.59 nM T51408 CV1FP0 24822817 EC50 = 0.46 nM T51408 CBRX49 24822819 EC50 = 0.54 nM T51408 CG13QX 24822970 EC50 = 32 nM T51408 CL4WP6 24822971 EC50 = 9.7 nM T51408 CWAO15 24822972 EC50 = 12 nM T51408 CVH1N4 24822974 EC50 = 2 nM T51408 CBS82N 24823127 EC50 = 1.1 nM T51408 C5NYS2 24823130 EC50 = 9.8 nM T51408 C0Q2ZB 24823131 EC50 = 17 nM T51408 CU3D5Q 24823134 EC50 = 4.3 nM T51408 C7US9I 24823292 EC50 = 0.81 nM T51408 CHUC65 24823294 EC50 = 0.3 nM T51408 CCF7Z8 24823296 EC50 = 0.34 nM T51408 C9MBA4 24823462 EC50 = 4 nM T51408 CHDE90 24823464 EC50 = 0.29 nM T51408 CJ9GR6 24823468 EC50 = 85 nM T51408 C5MS2U 24823470 EC50 = 18 nM T51408 CZ7UX0 24823624 EC50 = 4.6 nM T51408 CQ7C8J 24823626 EC50 = 5.5 nM T51408 C8Z3FQ 24823627 EC50 = 2.2 nM T51408 CE8N3Y 24823782 EC50 = 33 nM T51408 C0Q2KI 24824226 EC50 = 39 nM T51408 CT9QC7 24824227 EC50 = 61 nM T51408 C7FT4Z 24824228 EC50 = 100 nM T51408 C0EU5V 24824352 EC50 = 39 nM T51408 CR6N2C 24885648 Ki = 17 nM T51408 C1SFL2 24886595 Ki = 88 nM T51408 C08VXN 24893964 EC50 = 0.2512 nM T51408 CV5YU1 24893966 EC50 = 0.55 nM T51408 CYN9K4 24894127 EC50 = 5.2 nM T51408 C7FR5U 24894202 EC50 = 0.042 nM T51408 C9UV7P 24894315 EC50 = 0.5 nM T51408 C3W2AI 24894317 EC50 = 0.68 nM T51408 CGR30O 24894319 EC50 = 2.4 nM T51408 C5TR9W 24894323 EC50 = 0.21 nM T51408 C8ZG2O 24895192 EC50 = 2.1 nM T51408 CS1Q4X 24895194 EC50 = 30 nM T51408 C3Y6LC 24895196 EC50 = 8.1 nM T51408 CN1W9Y 24895259 EC50 = 0.26 nM T51408 C5AD3B 24895261 EC50 = 0.19 nM T51408 CW8V3F 24895263 EC50 = 0.035 nM T51408 CYG8J1 24895265 EC50 = 0.18 nM T51408 CLJ1U9 24895357 EC50 = 0.19 nM T51408 CULO78 24895359 EC50 = 0.79 nM T51408 CT7AM8 24895361 EC50 = 0.091 nM T51408 CA52PH 24895363 EC50 = 0.041 nM T51408 C76BAX 24895365 EC50 = 0.91 nM T51408 CF6SM4 24895557 EC50 = 0.21 nM T51408 CD26KH 24895559 EC50 = 0.32 nM T51408 C7YEW8 24895561 EC50 = 0.27 nM T51408 CG1D9Y 24895563 EC50 = 1.2 nM T51408 CT5HK9 24895565 EC50 = 0.16 nM T51408 CZ14LI 24895664 EC50 = 0.7 nM T51408 CE4K2V 24895667 EC50 = 2.4 nM T51408 CRN05D 24895669 EC50 = 0.062 nM T51408 C5OKI6 24895671 EC50 = 2.6 nM T51408 CIOG69 24895783 EC50 = 1.5 nM T51408 CQO97P 24895787 EC50 = 6 nM T51408 CLV98U 24895789 EC50 = 0.3 nM T51408 C5QLA9 24895791 EC50 = 0.31 nM T51408 C4BU6R 24936488 EC50 = 20 nM T51408 CH87SX 24936489 EC50 = 1.6 nM T51408 CIR69S 24936491 EC50 = 3.1 nM T51408 C75UCO 24936492 EC50 = 1 nM T51408 CRPN83 24936625 EC50 = 310 nM T51408 CT0ND6 24936626 EC50 = 0.02 nM T51408 CFZT09 24936627 EC50 = 2.9 nM T51408 CH7TO3 24936763 EC50 = 3.1 nM T51408 CKD63O 24936881 EC50 = 0.62 nM T51408 CTS43M 24936882 EC50 = 0.5 nM T51408 CWPZ46 24936883 EC50 = 97 nM T51408 C38LFU 24936885 EC50 = 0.14 nM T51408 CL91OF 24937013 EC50 = 2.2 nM T51408 C61SKD 24937014 EC50 = 1.7 nM T51408 CR13DN 24937016 EC50 = 33 nM T51408 CY4KV6 24937137 EC50 = 2 nM T51408 CA5HY0 24937140 IC50 = 162 nM T51408 CNP3A6 24937269 EC50 = 26 nM T51408 C9N1UV 24937387 Ki = 919 nM T51408 CZQH42 24937389 EC50 = 0.04 nM T51408 COLT89 24937390 EC50 = 7.8 nM T51408 C2H1AS 24949260 EC50 = 22 nM T51408 CX8N2G 24949262 EC50 = 7.1 nM T51408 C6CGT0 24949264 EC50 > 100 nM T51408 C1G4IU 24949414 EC50 = 49 nM T51408 CME8R0 24949416 EC50 = 10 nM T51408 CH6YJ7 24949418 EC50 = 2.8 nM T51408 CH0ZA8 24949420 EC50 = 9.6 nM T51408 CO2IH8 24949564 EC50 = 3.2 nM T51408 CMIA50 24949566 EC50 = 1.3 nM T51408 C2IN7M 24949568 EC50 = 1 nM T51408 CK2NO1 24949570 EC50 = 4.7 nM T51408 C4R8MP 24949572 EC50 = 4.1 nM T51408 CNV6F3 24949720 EC50 = 0.38 nM T51408 C12RTH 24949722 EC50 = 3.5 nM T51408 CIJ8T1 24949724 EC50 = 13 nM T51408 CK70NO 24949726 EC50 = 1.8 nM T51408 CIL04S 24949728 EC50 = 0.7 nM T51408 C16RWX 24949883 EC50 = 1.4 nM T51408 CFN26M 24949885 EC50 = 24 nM T51408 C9FWC3 24949887 EC50 = 37 nM T51408 C4Q1NP 24949889 EC50 = 4.5 nM T51408 CA5Q4V 24949891 EC50 = 1.47 nM T51408 C1VE2O 24950053 EC50 = 5.7 nM T51408 CH2R8Z 24950055 EC50 = 9 nM T51408 C8FY7G 24950057 EC50 = 16 nM T51408 CL5CM8 24950059 EC50 = 5.3 nM T51408 C8HMF4 24950061 EC50 = 3.2 nM T51408 C5VTD0 24950234 EC50 = 0.77 nM T51408 CQ80CT 24950236 EC50 = 0.78 nM T51408 CFZ85T 24950238 EC50 = 4.8 nM T51408 CJS80L 24950240 EC50 = 20 nM T51408 C3PB6N 24950242 EC50 = 3.6 nM T51408 CH2Q3D 24950401 EC50 = 1.8 nM T51408 CEU3F6 24950403 EC50 = 5.8 nM T51408 C2CD3O 24950405 EC50 = 29 nM T51408 CBX0L5 24950407 EC50 > 100 nM T51408 C6JXL4 24950409 EC50 = 2.4 nM T51408 CNR3Y4 24950560 EC50 = 38 nM T51408 C0M1XB 24950562 EC50 = 0.79 nM T51408 CH9U4B 24950564 EC50 = 28 nM T51408 CE0WB4 24950566 EC50 = 33 nM T51408 CMV2K0 24950568 EC50 = 0.85 nM T51408 CS7U5E 24950570 EC50 = 0.81 nM T51408 C5ZG2W 24950716 EC50 = 0.78 nM T51408 CLF4U7 24950718 EC50 = 2 nM T51408 C6FHK9 25071020 EC50 = 3.4 nM T51408 C2O0HZ 42609939 IC50 = 550 nM T51408 CAD31R 42611263 EC50 = 1584.89 nM T51408 C0FE1J 42625511 EC50 = 501.19 nM T51408 C7GK2I 42625513 EC50 = 1258.93 nM T51408 CE6IF3 42625515 EC50 = 794.33 nM T51408 C1BE8M 42625517 EC50 = 316.23 nM T51408 CL89KJ 42625587 EC50 = 158.49 nM T51408 CQ4O3V 42625588 EC50 = 2511.89 nM T51408 C9Q0OM 42625741 EC50 = 2511.89 nM T51408 CBN76E 42625743 EC50 = 1995.26 nM T51408 C6P3JN 42625821 EC50 = 630.96 nM T51408 C3JAT7 42625823 EC50 = 50.12 nM T51408 C4KE6Z 42625897 EC50 = 630.96 nM T51408 C6YR7G 42625898 EC50 = 316.23 nM T51408 CA2YO5 42639133 EC50 = 0.631 nM T51408 CRF79M 42639311 EC50 = 2.8 nM T51408 CP0D6A 42639314 EC50 = 0.38 nM T51408 C6I5KU 42639317 EC50 = 0.41 nM T51408 C7J1IV 42639487 EC50 = 0.33 nM T51408 CN6G7U 42639489 EC50 = 1.4 nM T51408 C1ORB7 42639491 EC50 = 0.5 nM T51408 CAJ05V 42639494 EC50 = 0.062 nM T51408 CCX13B 42639652 EC50 = 0.32 nM T51408 C9YFJ6 42639654 EC50 = 0.19 nM T51408 CFK5S7 42639656 EC50 = 0.0631 nM T51408 CK0X9P 42639806 EC50 = 18 nM T51408 C7IL9X 42639808 EC50 = 0.62 nM T51408 CTHM06 42639810 EC50 = 0.6 nM T51408 CTY09A 42639965 EC50 = 0.54 nM T51408 C97BUG 42639967 EC50 = 1 nM T51408 C4OU1Q 42639969 EC50 = 0.2 nM T51408 C9QLJ6 42640120 EC50 = 0.29 nM T51408 C21SKJ 42640122 EC50 = 0.1995 nM T51408 CB4Q8W 44126931 EC50 = 120 nM T51408 CWGQ16 44126933 EC50 = 240 nM T51408 CU8M4H 44127048 EC50 = 960 nM T51408 CXM3V6 44127050 EC50 = 740 nM T51408 CS0B5Z 44127052 EC50 = 360 nM T51408 C4H9TJ 44127054 EC50 = 1700 nM T51408 C2IC7Q 44127056 EC50 = 550 nM T51408 CAW50P 44127167 EC50 = 1500 nM T51408 CJ0S7Q 44127169 EC50 = 110 nM T51408 C53MWL 44127171 EC50 = 290 nM T51408 CX2VJ3 44127374 EC50 = 520 nM T51408 C8BRZ2 44127478 EC50 = 960 nM T51408 C6XMJ7 44127479 EC50 = 890 nM T51408 C6ULE4 44127480 EC50 = 1200 nM T51408 C1LWJ0 44127481 EC50 = 560 nM T51408 CCI02W 44127575 EC50 = 500 nM T51408 CL10EZ 44127677 EC50 = 650 nM T51408 C73XYH 44127678 EC50 = 140 nM T51408 CZ5FG8 44127679 EC50 = 83 nM T51408 CB1W9S 44127681 EC50 = 1700 nM T51408 CY39CN 44127782 EC50 = 470 nM T51408 C19VMJ 44186438 EC50 = 200 nM T51408 C2AV1K 44190762 IC50 = 4860 nM T51408 CLR40G 44219629 EC50 = 130 nM T51408 CZ2BO8 44219630 EC50 > 100000 nM T51408 CW7D8Q 44219641 EC50 = 30 nM T51408 C27AGX 44268214 EC50 = 600 nM T51408 C9D7RS 44268249 EC50 = 12 nM T51408 C4ML0P 44268253 EC50 = 1000 nM T51408 C5E2MI 44268254 EC50 = 440 nM T51408 CEF1D6 44268262 EC50 = 2000 nM T51408 CAY8L6 44268264 EC50 = 600 nM T51408 CNQ7X8 44268266 EC50 = 25 nM T51408 C72KSE 44268267 EC50 = 6000 nM T51408 CLR0X8 44268268 EC50 = 1.3 nM T51408 C9TB2F 44268273 EC50 = 54 nM T51408 C6NY3M 44268274 EC50 = 15 nM T51408 CGJT32 44268275 EC50 = 92 nM T51408 CZ3W8B 44268277 EC50 = 25 nM T51408 CLS1U8 44268281 EC50 = 4000 nM T51408 C6R8SP 44268295 EC50 = 60 nM T51408 C0UG8A 44268305 EC50 = 200 nM T51408 C2AJI5 44268308 EC50 = 4.3 nM T51408 CY6X8E 44268320 EC50 = 2.6 nM T51408 CCH34M 44268322 EC50 = 30 nM T51408 CAD4P0 44268324 EC50 = 4.8 nM T51408 CI91WY 44268327 EC50 = 1500 nM T51408 CMU89C 44268341 EC50 = 5.4 nM T51408 CS87PI 44268349 EC50 = 39 nM T51408 CB7F6R 44268352 EC50 = 110 nM T51408 CPNS03 44268358 EC50 = 58 nM T51408 C9JZ5T 44268365 EC50 = 62 nM T51408 CP2G7C 44268367 EC50 = 27 nM T51408 C1S3AB 44268464 EC50 = 11 nM T51408 C29IOC 44268470 EC50 = 6.8 nM T51408 CT3GL8 44268475 EC50 = 17 nM T51408 CI64OC 44268478 EC50 = 2.3 nM T51408 CU84BM 44268479 EC50 = 2.6 nM T51408 CQY09P 44268482 EC50 = 5 nM T51408 CRV1T3 44268495 EC50 = 1 nM T51408 CU21DW 44268496 EC50 = 1.2 nM T51408 C2HDU8 44268497 EC50 = 4.6 nM T51408 CWG2Q7 44268498 EC50 = 10 nM T51408 C4D1OQ 44268509 EC50 = 1.4 nM T51408 C3YGB4 44268520 EC50 = 1 nM T51408 C5TZ8J 44268534 EC50 = 1.1 nM T51408 CS73JY 44268539 EC50 = 1.2 nM T51408 CN8P2B 44268556 EC50 = 0.7 nM T51408 CES3Y9 44268563 EC50 = 1.4 nM T51408 CY5J3N 44268568 EC50 = 5.2 nM T51408 CREN46 44268569 EC50 = 6.6 nM T51408 C0BR2A 44268570 EC50 = 2.1 nM T51408 C9H1IF 44268571 EC50 = 1.9 nM T51408 CBZ7N6 44268572 EC50 = 2.4 nM T51408 C2LYD1 44268604 EC50 = 2.8 nM T51408 CD7UZ0 44268605 EC50 = 1.1 nM T51408 CF3VU1 44268632 EC50 = 1.4 nM T51408 CW7A6K 44280795 EC50 = 87 nM T51408 CR8D7Y 44280858 EC50 = 54 nM T51408 C4JLV9 44280860 EC50 = 32 nM T51408 C49FOW 44280903 EC50 = 5 nM T51408 CM6C4J 44280904 EC50 = 2 nM T51408 CJ1B9Z 44280957 EC50 = 120 nM T51408 CM9R8D 44281037 EC50 > 100 nM T51408 CPO25L 44281073 EC50 = 75 nM T51408 CI4NE5 44281074 EC50 = 66 nM T51408 CG7A5O 44281097 EC50 = 12 nM T51408 CS84VC 44281218 EC50 = 3 nM T51408 CIPT87 44281219 EC50 = 8 nM T51408 C1S3HD 44281255 EC50 = 29 nM T51408 CZT1Q6 44281276 EC50 = 35 nM T51408 COB42G 44281277 EC50 = 39 nM T51408 C28KLB 44281344 EC50 = 31 nM T51408 C65JLA 44281371 EC50 = 8 nM T51408 CD78QG 44281372 EC50 = 7 nM T51408 CBNZ27 44281384 EC50 = 6 nM T51408 CG3D5J 44281395 EC50 = 6 nM T51408 CBL4F1 44281396 EC50 = 4 nM T51408 CO9F8Q 44281400 EC50 = 4 nM T51408 CT0XW9 44281407 EC50 = 11 nM T51408 CK3Z4L 44281408 EC50 = 10 nM T51408 C7P3WY 44281424 EC50 = 10 nM T51408 CIO1V4 44281425 EC50 = 190 nM T51408 CJU5O2 44281467 EC50 = 79 nM T51408 CI1C5Q 44281468 EC50 = 15 nM T51408 CTL1G7 44281469 EC50 = 12 nM T51408 CEN7H9 44281470 EC50 = 8 nM T51408 CC90RN 44281530 EC50 = 2 nM T51408 CLXI95 44281531 EC50 = 3 nM T51408 C0DG5M 44285225 EC50 = 230 nM T51408 CNO3I4 44285226 EC50 = 34 nM T51408 C7L5MN 44285529 EC50 = 26 nM T51408 CUF3O2 44285634 EC50 = 12 nM T51408 CTIA64 44285685 EC50 > 100 nM T51408 C0JY4C 44285692 EC50 = 76 nM T51408 CPQ16U 44286964 EC50 = 2640 nM T51408 CKL84D 44286965 EC50 = 750 nM T51408 C2IJ9G 44286980 Ki = 19900 nM T51408 CPN74V 44286983 EC50 = 1610 nM T51408 CE5GK6 44287268 EC50 = 610 nM T51408 CD0E2S 44287321 Ki = 11100 nM T51408 CA72HF 44287337 EC50 = 1610 nM T51408 C53RQT 44298256 EC50 = 13 nM T51408 C82TAV 44298288 EC50 = 0.9 nM T51408 C0ICR9 44298290 EC50 = 8.1 nM T51408 COTF72 44298306 EC50 = 55 nM T51408 CIJ6H2 44298315 EC50 = 31 nM T51408 CDCP96 44298497 EC50 = 2.4 nM T51408 CNK60M 44298515 EC50 = 5.1 nM T51408 CZHU81 44298516 EC50 = 3.2 nM T51408 CJ1X0Z 44298533 EC50 = 0.93 nM T51408 CRD69E 44298695 EC50 = 7 nM T51408 CSKD26 44298718 EC50 = 88 nM T51408 CBW06V 44298728 EC50 = 6.9 nM T51408 CVN75C 44298731 EC50 = 0.73 nM T51408 C67YCD 44298752 EC50 = 47 nM T51408 CO9BE8 44298761 EC50 = 55 nM T51408 CD51GN 44298769 EC50 = 5.5 nM T51408 CE01UQ 44298781 EC50 = 18 nM T51408 CUK01S 44298787 EC50 = 0.8 nM T51408 CAP4B0 44298804 EC50 = 0.65 nM T51408 CFRN96 44298821 EC50 = 3.7 nM T51408 C40OYU 44298822 EC50 = 5 nM T51408 C19XHR 44298823 EC50 = 1.3 nM T51408 CSW8G0 44298843 EC50 = 1.6 nM T51408 CQID30 44298849 EC50 = 1.8 nM T51408 C8FL6R 44298850 EC50 = 1.7 nM T51408 CHJR57 44298851 EC50 = 1 nM T51408 C2GBS7 44298852 EC50 = 1.2 nM T51408 C6GD9N 44301617 EC50 = 1.2 nM T51408 CI0OY1 44301618 EC50 = 9.5 nM T51408 C4P1OD 44301764 EC50 = 51 nM T51408 CCH74I 44301803 EC50 = 6.2 nM T51408 C3T9OF 44301804 EC50 = 22 nM T51408 CY63AQ 44301805 EC50 = 40 nM T51408 CA3VZ2 44301806 EC50 = 2.7 nM T51408 C2OJ3N 44301818 EC50 = 45 nM T51408 CNZ68T 44301819 EC50 = 2.4 nM T51408 CMFW56 44301831 EC50 = 26 nM T51408 CJB9L8 44301832 EC50 = 10 nM T51408 C4DZ6V 44301842 EC50 = 2 nM T51408 CW02XN 44301843 EC50 = 33 nM T51408 C6P8UW 44301866 EC50 = 9.8 nM T51408 C8T7OB 44301867 EC50 = 45 nM T51408 CS4ET3 44301880 EC50 = 9.1 nM T51408 CM4G9Z 44301881 EC50 = 5.8 nM T51408 C6VDZ8 44301886 EC50 = 50 nM T51408 C08SKL 44301979 EC50 = 7.3 nM T51408 C8EGA1 44302005 EC50 = 4.9 nM T51408 C9J6RY 44303192 EC50 = 56 nM T51408 CN0DE9 44303198 EC50 = 7.8 nM T51408 C5JS0C 44303416 EC50 < 300 nM T51408 CF5Q7X 44303556 EC50 = 0.06 nM T51408 CA4BQ1 44306956 EC50 = 24 nM T51408 C70GLV 44306959 EC50 = 13 nM T51408 C9HL3E 44306979 EC50 = 30 nM T51408 C75OJI 44306985 EC50 = 26 nM T51408 CH58SX 44306991 EC50 = 43 nM T51408 C0XI5A 44306992 EC50 = 400 nM T51408 CN23SP 44307007 EC50 = 85 nM T51408 C4LRJ3 44307063 EC50 = 22 nM T51408 CYI2V9 44307064 EC50 = 73 nM T51408 C7KWF2 44307065 EC50 = 18 nM T51408 CF01WZ 44307085 EC50 = 3.3 nM T51408 C3H9QV 44307113 EC50 = 120 nM T51408 CC4IL0 44307144 EC50 = 3.8 nM T51408 CBC1J6 44307148 EC50 = 6.4 nM T51408 CK0WG5 44307166 EC50 = 18 nM T51408 CLB56U 44307186 EC50 = 23 nM T51408 CYX08L 44307196 EC50 = 43 nM T51408 CNCV21 44307205 EC50 = 6 nM T51408 C5Q4MP 44307333 EC50 = 22 nM T51408 CVK8S0 44307340 EC50 = 26 nM T51408 C1RYI9 44307343 EC50 = 7 nM T51408 CK1P5Z 44307378 EC50 = 32 nM T51408 CV1Z0F 44307379 EC50 = 32 nM T51408 C5NIP7 44307396 EC50 = 5 nM T51408 C9G4UO 44309272 EC50 = 5 nM T51408 CM4KI1 44309305 EC50 = 1100 nM T51408 C6C1XR 44309320 EC50 = 360 nM T51408 CRE39G 44309322 EC50 = 850 nM T51408 C8YIN9 44309363 EC50 = 120 nM T51408 C8HK0V 44309512 EC50 > 2000 nM T51408 CKWA37 44309523 EC50 = 30 nM T51408 C6O7IR 44309633 EC50 = 920 nM T51408 CMJX34 44309649 EC50 = 55 nM T51408 CM70FY 44309650 EC50 > 2000 nM T51408 C1LBM4 44311101 EC50 = 820 nM T51408 CP96BD 44311119 EC50 = 2200 nM T51408 C20IGU 44311370 EC50 = 1000 nM T51408 C1QTH9 44311371 EC50 = 2000 nM T51408 CCQ2H4 44311447 EC50 = 560 nM T51408 CVN87R 44311597 EC50 = 290 nM T51408 CP5W8S 44311756 EC50 = 1100 nM T51408 CY9NW5 44311757 EC50 = 7900 nM T51408 C9XMY7 44311778 EC50 = 4700 nM T51408 CVKS51 44311779 EC50 = 400 nM T51408 CFHD64 44312269 Ki = 36500 nM T51408 CVX04Z 44312421 Ki = 390 nM T51408 CF3H5U 44312924 EC50 = 27 nM T51408 CY4K0A 44312949 EC50 = 7 nM T51408 C3L4PJ 44313090 EC50 = 4 nM T51408 CL2UV6 44313150 EC50 = 360 nM T51408 CPA5B7 44313161 EC50 = 10 nM T51408 CV8J4A 44331302 EC50 = 5 nM T51408 C97IJY 44331346 EC50 = 6 nM T51408 C0RDZ3 44331351 EC50 = 31 nM T51408 CIFO93 44331425 EC50 = 10 nM T51408 C5Y8GN 44331426 EC50 = 6 nM T51408 CU4EQ5 44331443 EC50 = 31 nM T51408 CWE69G 44331444 EC50 = 27 nM T51408 CCA29H 44331530 EC50 = 306 nM T51408 CZQ14C 44331551 EC50 = 870 nM T51408 C3OIA6 44331553 EC50 = 290 nM T51408 CI17GW 44331766 EC50 = 187 nM T51408 C4X8MT 44331791 EC50 = 319 nM T51408 C8JKE3 44333524 Ki = 210 nM T51408 CEYN93 44333531 Ki = 26 nM T51408 C75VMA 44333536 Ki = 9 nM T51408 C8N1MZ 44333551 Ki = 300 nM T51408 CIA6F5 44333588 Ki = 81 nM T51408 C10NXD 44333605 Ki = 220 nM T51408 C8NW6Z 44333651 Ki = 38 nM T51408 C2Y3TA 44333696 Ki = 11 nM T51408 CS52CU 44333716 Ki = 4300 nM T51408 CE12RV 44333719 Ki = 1550 nM T51408 C8GV9C 44333726 Ki = 81 nM T51408 C6NQH8 44333733 Ki = 5800 nM T51408 CF3G0I 44333734 Ki = 320 nM T51408 C08KVO 44333737 Ki = 12700 nM T51408 CG62ZM 44333738 Ki = 550 nM T51408 CAK7L6 44333757 Ki = 15 nM T51408 CA9Q8I 44333758 Ki = 25 nM T51408 C4PM7D 44333761 Ki = 3700 nM T51408 C4HVR2 44333764 Ki = 2800 nM T51408 CK6O7D 44333790 Ki = 980 nM T51408 C53HRZ 44333795 Ki = 570 nM T51408 CIKR37 44333796 Ki = 230 nM T51408 CK0DU4 44333797 Ki = 49000 nM T51408 C91RKL 44333802 Ki = 70 nM T51408 CUN2S1 44333818 Ki = 1500 nM T51408 CWKI43 44333828 Ki = 11000 nM T51408 C47XRV 44333830 Ki = 990 nM T51408 CD8WT1 44333846 Ki = 43 nM T51408 CC1B2U 44333847 Ki = 69 nM T51408 C7EPJ2 44333853 Ki = 84 nM T51408 CZJ2N8 44333864 Ki = 2400 nM T51408 CRU2N4 44333890 Ki = 147 nM T51408 C1CZD5 44333920 Ki = 85 nM T51408 COJ6B1 44333923 Ki = 480 nM T51408 CLH92K 44333932 Ki = 20 nM T51408 C83LDW 44333968 Ki = 2 nM T51408 CF9E4B 44334123 Ki = 1100 nM T51408 CQE1H6 44334131 Ki = 3300 nM T51408 CZF1C0 44334144 Ki = 836 nM T51408 C2I6EM 44334164 Ki = 320 nM T51408 CG8O7B 44334231 Ki = 210 nM T51408 C5BX2N 44335497 EC50 = 160 nM T51408 CD7ZV4 44335498 EC50 = 38 nM T51408 C9UE7G 44335499 EC50 = 56 nM T51408 CDS5L1 44335534 EC50 = 1.6 nM T51408 C7MC1U 44335548 EC50 = 1.4 nM T51408 CY7LH9 44335560 EC50 = 100 nM T51408 C6IA8P 44335562 EC50 = 18 nM T51408 CLE91U 44335572 EC50 = 77 nM T51408 C4B8OE 44335588 EC50 = 67 nM T51408 C17PHB 44335589 EC50 = 27 nM T51408 C7A4UT 44335603 EC50 = 18 nM T51408 CFX90I 44335618 EC50 = 68 nM T51408 C14ILU 44335628 EC50 = 150 nM T51408 CX8QZ4 44335651 EC50 = 49 nM T51408 C03GDI 44335663 EC50 = 67 nM T51408 CM0XE7 44336180 EC50 = 30 nM T51408 CNW2Y0 44336319 EC50 = 5 nM T51408 CF9V7S 44344526 Ki = 8200 nM T51408 C08EHN 44344575 Ki = 490 nM T51408 CDYV51 44344578 Ki = 3100 nM T51408 C49RHY 44344592 Ki = 17 nM T51408 CUG5R9 44344593 Ki = 142 nM T51408 CS03NV 44344618 Ki = 61 nM T51408 CVP5L1 44344619 Ki = 71 nM T51408 C5DGE0 44344649 Ki = 14 nM T51408 CQ23SJ 44344650 Ki = 19 nM T51408 CAFK40 44344656 Ki = 20 nM T51408 CO03VN 44344670 Ki = 11 nM T51408 CEZ4D3 44344671 Ki = 23 nM T51408 C6RYQ2 44344674 Ki = 340 nM T51408 C3MI7R 44344701 Ki = 950 nM T51408 C9AR0T 44344713 Ki = 190 nM T51408 CATV47 44344714 Ki = 400 nM T51408 CR28MU 44344757 Ki = 2910 nM T51408 CWNS24 44344758 Ki = 2200 nM T51408 C3XU2F 44344787 Ki = 380 nM T51408 CPL96K 44344806 Ki = 28 nM T51408 C6YRX1 44344819 Ki = 46 nM T51408 C2EDG5 44344820 Ki = 51 nM T51408 CQ64AZ 44344828 Ki = 47 nM T51408 CXV9Q2 44344829 Ki = 17 nM T51408 CV79WH 44344870 Ki = 24 nM T51408 CS76IR 44344909 Ki = 260 nM T51408 CCZ86G 44344910 Ki = 520 nM T51408 CG24EN 44344911 Ki = 370 nM T51408 C48AHQ 44344912 Ki = 115 nM T51408 CW6LN8 44344960 Ki = 44 nM T51408 CSHW18 44345040 Ki = 370 nM T51408 COQ8L1 44345048 Ki = 450 nM T51408 C9Y4AL 44345049 Ki = 1800 nM T51408 C6N3XK 44345317 IC50 < 1000 nM T51408 C4PU1O 44349588 EC50 = 5.3 nM T51408 CS1L9V 44349629 EC50 = 130 nM T51408 C6WP1E 44349646 EC50 = 59 nM T51408 CZK46C 44369602 EC50 = 316.23 nM T51408 C3M7BC 44377315 EC50 = 2.5 nM T51408 CS6C8L 44377316 EC50 = 5.8 nM T51408 CJ4DO1 44377483 EC50 = 220 nM T51408 CEW6J9 44377513 EC50 = 15 nM T51408 C8DYK5 44377514 EC50 = 5.4 nM T51408 CRB49F 44377517 EC50 = 21 nM T51408 C3XLD1 44377636 EC50 = 9.5 nM T51408 C3BQ1X 44377637 EC50 = 4.4 nM T51408 CHB6Q2 44377650 EC50 = 13 nM T51408 CNEO30 44377665 EC50 = 67 nM T51408 CKI9O8 44377677 EC50 = 85 nM T51408 CQEA58 44377687 EC50 = 20 nM T51408 C49FSC 44377753 EC50 = 2.6 nM T51408 CW42ZY 44377754 EC50 = 1.6 nM T51408 C04XMY 44377755 EC50 = 25 nM T51408 C02ZPF 44377957 EC50 = 37 nM T51408 CESH03 44385716 EC50 = 75 nM T51408 C98GUQ 44385820 EC50 = 9 nM T51408 C7IW9X 44385888 EC50 = 2 nM T51408 C47PAS 44386051 EC50 = 940 nM T51408 CG5I3L 44386136 EC50 = 400 nM T51408 CN25BP 44386368 EC50 = 9 nM T51408 CA0FJ7 44386369 EC50 = 1 nM T51408 CXN97Q 44386374 EC50 = 6 nM T51408 CG2F6I 44386630 EC50 = 10 nM T51408 C8R4CT 44386631 EC50 = 3 nM T51408 CQ3OE6 44392175 EC50 = 1 nM T51408 C0S9HV 44392181 EC50 = 1.1 nM T51408 C82SPF 44392190 EC50 = 13 nM T51408 CE2M3X 44392212 EC50 = 1.6 nM T51408 CDF75J 44392215 EC50 = 2.5 nM T51408 CB9NO4 44392223 EC50 = 74 nM T51408 CO43RV 44392228 EC50 = 2.1 nM T51408 C96SHC 44392230 EC50 = 1.5 nM T51408 C5BEG3 44392238 EC50 = 22 nM T51408 C37GEF 44392240 EC50 = 8.3 nM T51408 CYEF45 44392255 EC50 = 4.9 nM T51408 C0CBD4 44392457 EC50 = 1.2 nM T51408 CES46V 44392480 EC50 = 9 nM T51408 CXO92R 44392490 EC50 = 160 nM T51408 CH21LQ 44392499 EC50 = 100 nM T51408 CHIC83 44392508 EC50 = 15 nM T51408 C7D8AU 44392519 EC50 = 11 nM T51408 CMH6N4 44392534 EC50 = 3.2 nM T51408 C7QJN5 44392542 EC50 = 2.9 nM T51408 CND67K 44392552 EC50 = 0.54 nM T51408 CS3H7D 44392558 EC50 = 36 nM T51408 C9GQ5B 44392559 EC50 = 52 nM T51408 CCZQ48 44392566 EC50 = 17 nM T51408 C65AEC 44392569 EC50 = 32 nM T51408 C83OKR 44392575 EC50 = 10 nM T51408 CADQ67 44392577 EC50 = 6.5 nM T51408 CI4J7L 44396488 EC50 = 1.3 nM T51408 CY46LP 44396509 EC50 = 2 nM T51408 CB37RE 44396513 EC50 = 0.51 nM T51408 C6HQL1 44396521 EC50 = 4.3 nM T51408 CE1MS4 44396530 EC50 = 0.59 nM T51408 C2YP6O 44396531 EC50 = 0.28 nM T51408 CLYG39 44396532 EC50 = 0.88 nM T51408 CJ75RF 44396559 EC50 = 1 nM T51408 CN7HX8 44396568 EC50 = 1.7 nM T51408 C0O6RE 44396574 EC50 = 2.8 nM T51408 C2DOA1 44396577 EC50 = 0.76 nM T51408 CHXA19 44396596 EC50 = 0.55 nM T51408 C27VFN 44396615 EC50 = 2 nM T51408 CD6A7V 44396616 EC50 = 25 nM T51408 C5HO7D 44396623 EC50 = 8.4 nM T51408 CW7B5D 44396625 EC50 = 1 nM T51408 CPR37V 44396632 EC50 = 48 nM T51408 COS8K3 44396654 EC50 = 2.4 nM T51408 CZ71YN 44396659 EC50 = 1.7 nM T51408 CT07OY 44396671 EC50 = 6.7 nM T51408 C4ABS7 44396673 EC50 = 3 nM T51408 CSB60T 44396675 EC50 = 0.94 nM T51408 CA52MR 44396678 EC50 = 21 nM T51408 C7RJ5T 44396681 EC50 = 18 nM T51408 CW4OR6 44396715 EC50 = 0.26 nM T51408 C4BXY6 44396729 EC50 = 0.31 nM T51408 C6ZND4 44396730 EC50 = 7.6 nM T51408 CRY62C 44396736 EC50 = 0.64 nM T51408 C4WO2Y 44396737 EC50 = 1.2 nM T51408 C6CZX4 44396738 EC50 = 1.1 nM T51408 CYS43A 44396739 EC50 = 13 nM T51408 CUO7X8 44396779 EC50 = 0.87 nM T51408 CYV72Q 44396784 EC50 = 20 nM T51408 C53GBI 44396798 EC50 = 0.47 nM T51408 CPZ8B0 44402687 EC50 = 9.8 nM T51408 CV7EO3 44402688 EC50 = 12 nM T51408 C2M7CT 44402689 EC50 = 51 nM T51408 CLFM57 44402690 EC50 = 26 nM T51408 C3FWK4 44402691 EC50 = 2 nM T51408 C9U2AI 44402692 EC50 = 5.8 nM T51408 C3RY0M 44402693 EC50 = 7.3 nM T51408 C5XUE0 44402694 EC50 = 2.7 nM T51408 C7UJ3L 44402695 EC50 = 9.5 nM T51408 CG5Q6K 44402728 EC50 = 9.1 nM T51408 C7ZSO2 44402729 EC50 = 40 nM T51408 CYJD67 44402730 EC50 = 22 nM T51408 CMW70L 44402731 EC50 = 7.1 nM T51408 C13GXE 44402732 EC50 = 1.2 nM T51408 C7AD6X 44402733 EC50 = 2.4 nM T51408 CKY7X1 44402734 EC50 = 45 nM T51408 CCT7B6 44402735 EC50 = 45 nM T51408 CN67IT 44402803 EC50 = 6.2 nM T51408 CV63NB 44402821 EC50 = 10 nM T51408 CR24VU 44402822 EC50 = 50 nM T51408 C01IDH 44402823 EC50 = 33 nM T51408 CLOF83 44402838 EC50 = 33 nM T51408 CXW84E 44402839 EC50 = 5 nM T51408 CSA2X5 44419254 EC50 = 11.7 nM T51408 CG5XU6 44419315 EC50 = 5.2 nM T51408 C4ABS0 44419316 EC50 = 5.4 nM T51408 CQ89AE 44419324 EC50 = 5.2 nM T51408 CFG74O 44419332 EC50 = 7.1 nM T51408 C5YBA0 44423639 Ki > 100000 nM T51408 C3XR8N 44423640 Ki = 22000 nM T51408 C45ISV 44423641 Ki > 50000 nM T51408 CK1XO7 44423643 Ki = 10100 nM T51408 CD72TX 44423644 Ki = 21800 nM T51408 C34MXL 44423645 Ki = 2485 nM T51408 C7IAO1 44423646 Ki = 10700 nM T51408 CN8G6D 44441226 EC50 = 15.85 nM T51408 C4Q1JB 44441227 EC50 = 15.85 nM T51408 CC34NU 44441228 EC50 = 6.31 nM T51408 CE34HD 44441229 EC50 = 0.7943 nM T51408 CXE23W 44441230 EC50 = 1.585 nM T51408 CZ96SJ 44441231 EC50 = 1.995 nM T51408 CTWM30 44441232 EC50 = 1.259 nM T51408 CA8E5H 44441233 EC50 = 3.981 nM T51408 CP2H0M 44441234 EC50 = 0.3162 nM T51408 CZ2K7C 44441235 EC50 = 0.3981 nM T51408 CR9B1F 44441236 EC50 = 1.259 nM T51408 CK57LZ 44444149 Ki = 7 nM T51408 C2QM7K 44444151 Ki = 93 nM T51408 CX5S9F 44444152 Ki = 120000 nM T51408 C6MFP8 44444153 EC50 = 24.4 nM T51408 C1QZW9 44444154 EC50 = 12 nM T51408 CJNU87 44444156 Ki = 270 nM T51408 CMG35K 44444157 Ki = 200 nM T51408 C8IF1O 44444158 Ki = 1700 nM T51408 C3M5QK 44444159 Ki = 15000 nM T51408 CX8GL7 44444160 Ki = 360 nM T51408 C15OUP 44444162 Ki = 5 nM T51408 C71SAB 44444163 Ki = 3 nM T51408 CR8ST7 44444164 Ki = 3700 nM T51408 CE5HX3 44444165 Ki = 880 nM T51408 CGDZ68 44444166 EC50 = 13.9 nM T51408 C9OIT6 44444167 EC50 = 14 nM T51408 C51KOV 44444168 Ki = 160 nM T51408 CG2QI4 44444169 EC50 = 12.3 nM T51408 C58UHL 44444170 Ki = 1100 nM T51408 CUAN40 44444171 EC50 = 2.7 nM T51408 CVQ59T 44444172 EC50 = 268.1 nM T51408 C60YDC 44444173 EC50 = 6.6 nM T51408 C1IB7H 44444175 EC50 = 17.6 nM T51408 CZ0VJ5 44444176 EC50 = 8.3 nM T51408 CD74SN 44444179 Ki = 133 nM T51408 C76QWZ 44444181 Ki = 340 nM T51408 CL18KR 44444184 Ki = 170 nM T51408 C5TM3W 44444185 Ki = 9 nM T51408 C16XQT 44444187 Ki = 31 nM T51408 C6PS3A 44444188 Ki = 390 nM T51408 CZAK23 44444189 Ki = 59 nM T51408 C9A3KP 44444191 Ki = 7 nM T51408 CA08VR 44444193 Ki = 29 nM T51408 CNS8K2 44444195 Ki = 12 nM T51408 C9FU0M 44444356 EC50 = 1360 nM T51408 CTCN06 44444359 EC50 = 2250 nM T51408 CB2HV4 44444361 EC50 = 2740 nM T51408 CNG2B4 44444363 EC50 = 1190 nM T51408 C8E2VD 44444365 EC50 = 4490 nM T51408 CZ2QL6 44444367 EC50 = 230 nM T51408 CYG1L2 44444369 EC50 = 130 nM T51408 CLO4K3 44444370 EC50 = 490 nM T51408 C0SA8C 44444378 EC50 = 120 nM T51408 C9QP8S 44444393 EC50 = 606 nM T51408 CZL97F 44455426 Ki > 10000 nM T51408 C12XGE 44456400 Ki > 10000 nM T51408 C1A6ZC 44457929 EC50 = 6.3 nM T51408 C7O0IE 44458134 EC50 = 30 nM T51408 C68NOT 44461468 EC50 = 100 nM T51408 CDZ56W 44461485 EC50 = 100 nM T51408 CM5ZH4 44461486 EC50 = 6 nM T51408 C2GZ3R 44461488 EC50 = 130 nM T51408 C1L6GN 44461489 EC50 = 18 nM T51408 CVC1K4 44461490 EC50 = 15 nM T51408 CABF14 44461496 EC50 = 5.4 nM T51408 CQ8UE4 44461716 EC50 = 60 nM T51408 C4TMP7 44461717 EC50 = 81 nM T51408 C39FRG 44461718 EC50 = 3.4 nM T51408 CM4F7J 44461719 EC50 = 14 nM T51408 C2QK4J 44472590 EC50 = 0.9 nM T51408 CQ8C3F 44472591 EC50 = 1.7 nM T51408 CC2TA5 44472592 EC50 = 3.9 nM T51408 CWN95E 44472610 EC50 = 4.8 nM T51408 C1H2ZT 44472612 EC50 = 2.2 nM T51408 C9G5ID 44472613 EC50 = 4.3 nM T51408 C5N4KE 44472633 EC50 = 0.62 nM T51408 CEH82X 44472636 EC50 = 0.18 nM T51408 CMH3J4 44472637 EC50 = 0.67 nM T51408 CC6G0Z 44517692 EC50 = 100 nM T51408 C5BYX7 44517694 EC50 = 160 nM T51408 CY8PO3 44517696 EC50 = 200 nM T51408 CS8G3O 44560739 EC50 = 7.4 nM T51408 CE18ZY 44560791 EC50 = 0.49 nM T51408 C7V8EF 44560792 EC50 = 0.099 nM T51408 CMP8T6 44560793 EC50 = 0.064 nM T51408 CP36SU 44560794 EC50 = 0.069 nM T51408 C9P7BS 44565907 EC50 = 0.68 nM T51408 CP0JB5 44565908 EC50 = 0.1259 nM T51408 CAF8L7 44565931 EC50 = 0.029 nM T51408 CDUZ13 44565932 EC50 = 0.08 nM T51408 CBD52U 44574651 EC50 > 100000 nM T51408 CSGI84 44574685 EC50 > 100000 nM T51408 CIF02K 44574686 EC50 > 100000 nM T51408 C4PN5S 44574687 EC50 > 100000 nM T51408 C6BVQ7 44574688 EC50 > 100000 nM T51408 C6UTI8 44574720 EC50 > 100000 nM T51408 C0RB7H 44574721 EC50 = 390 nM T51408 C56UZO 44574722 EC50 = 310 nM T51408 CVP31K 44574723 EC50 = 55 nM T51408 CM53PL 44574757 EC50 = 200 nM T51408 CLG2N1 44574758 EC50 = 510 nM T51408 C6E2SN 44574759 EC50 > 100000 nM T51408 CIS5B4 44574825 EC50 > 100000 nM T51408 CK2H8G 44574826 EC50 = 280 nM T51408 CU7H5I 44574827 EC50 = 74 nM T51408 C9GZ3R 44574867 EC50 = 71 nM T51408 CL7SJ3 44574868 EC50 = 69 nM T51408 C9HE8U 44574913 EC50 > 100000 nM T51408 CO3V6F 44574978 EC50 = 120 nM T51408 CKE82M 44579649 EC50 = 56 nM T51408 C0OHE7 44579650 EC50 = 12 nM T51408 CS92ZG 44579651 EC50 = 1.9 nM T51408 CA5O2G 44579925 EC50 = 9.5 nM T51408 C90FXY 44579940 EC50 = 6.5 nM T51408 CUZ85X 44579941 EC50 = 6.6 nM T51408 CLU26M 44579964 EC50 = 60 nM T51408 C81ALE 44579965 EC50 = 14 nM T51408 C6LV4K 44579966 EC50 = 9.4 nM T51408 CZL47Y 44580009 EC50 = 13 nM T51408 C86TQI 44580010 EC50 = 11 nM T51408 C8C0FP 44580011 EC50 = 7.2 nM T51408 CTE0P6 44580039 EC50 = 8.6 nM T51408 CZ3OG8 44580040 EC50 = 4.6 nM T51408 C5YB0H 44580041 EC50 = 21 nM T51408 CBH97I 44580042 EC50 = 31 nM T51408 CRCH48 44582675 Ki > 10000 nM T51408 CEJ4R8 44582676 Ki > 10000 nM T51408 C5QB4K 44582678 Ki > 10000 nM T51408 C01RCI 44582705 Ki > 10000 nM T51408 C3L5ER 44583033 EC50 = 7 nM T51408 CXD63G 44589133 EC50 = 883 nM T51408 CS08ED 44589400 IC50 = 1180 nM T51408 CX5O1N 44589401 IC50 = 1760 nM T51408 CJ0D9X 44591506 EC50 = 0.19 nM T51408 C32HSU 44591507 EC50 = 0.066 nM T51408 CWQ2K4 44591508 EC50 = 0.035 nM T51408 C7CM3S 45101537 EC50 = 0.16 nM T51408 C07LMT 45267257 EC50 = 340 nM T51408 C7OTL6 45267631 EC50 = 0.82 nM T51408 C5P2KR 45268128 EC50 = 460 nM T51408 C7NC2T 45268136 EC50 = 100 nM T51408 C9SIW5 45268516 EC50 = 0.26 nM T51408 C7GPS1 45269025 EC50 = 320 nM T51408 C2D7EA 45269373 EC50 = 6 nM T51408 CEA21T 45269853 EC50 = 410 nM T51408 C5EO1Y 45270197 EC50 = 1.2 nM T51408 CH2Y3X 45270673 EC50 = 570 nM T51408 CW2FT8 45270680 EC50 = 440 nM T51408 C43UZN 45270690 EC50 = 340 nM T51408 CCZ10H 45270697 EC50 = 270 nM T51408 CGTY98 45271036 EC50 = 0.044 nM T51408 CG2L0D 45271492 EC50 = 330 nM T51408 CK48MV 45271517 EC50 = 230 nM T51408 C13VYN 45271518 EC50 = 170 nM T51408 CMU01B 45271523 EC50 = 600 nM T51408 C0QOW1 45271886 EC50 = 0.1 nM T51408 CS27QE 45272430 EC50 = 230 nM T51408 CL76SG 45272431 EC50 = 470 nM T51408 C07GYE 45272758 EC50 = 28 nM T51408 CBKW49 45273268 EC50 = 310 nM T51408 C6GW4V 45273276 EC50 = 550 nM T51408 CH10SC 45273280 EC50 = 470 nM T51408 CM5H4D 45280021 EC50 = 66 nM T51408 CPJB52 45280075 EC50 = 17 nM T51408 CV0JK1 45380469 EC50 = 70 nM T51408 C6QES8 45380471 EC50 = 3.9 nM T51408 CZ73IE 45381852 EC50 = 14 nM T51408 CNI72R 45381932 EC50 = 13 nM T51408 C8WG5T 45381933 EC50 = 64 nM T51408 C7NA1H 46832227 EC50 = 12589.25 nM T51408 CNA42V 46832232 EC50 = 5.012 nM T51408 CN7MG5 46832505 EC50 = 39.81 nM T51408 CJ5B4A 46832507 EC50 = 316.23 nM T51408 CW0JV6 46832509 EC50 = 79.43 nM T51408 C7TN0H 46832510 EC50 = 794.33 nM T51408 C04XPW 46832798 EC50 = 7.943 nM T51408 CQ1BJ4 46832804 EC50 = 398.11 nM T51408 C6VS1A 46833102 EC50 = 125.89 nM T51408 CSYQ43 46833103 EC50 = 63.1 nM T51408 CQ3TM8 46845697 EC50 = 37 nM T51408 CJV15G 46845698 EC50 = 73 nM T51408 C0DB5H 46845699 EC50 = 76 nM T51408 C2D6ZI 46881527 EC50 = 297 nM T51408 CIP0H2 46881528 EC50 = 95 nM T51408 CZ0PU9 46881529 EC50 = 225 nM T51408 CTV6U8 46881530 EC50 = 8.8 nM T51408 CFA38Z 46881531 EC50 = 19 nM T51408 CIJU02 46881573 EC50 = 48 nM T51408 C4YNT0 46881574 EC50 = 14 nM T51408 CV5R2L 46881575 EC50 = 24 nM T51408 CULH08 46881576 EC50 = 21 nM T51408 CYLF92 46881614 EC50 = 693 nM T51408 CT56SD 46881615 EC50 = 22 nM T51408 CLB86Z 46881616 EC50 = 103 nM T51408 CJ1VO4 46881617 EC50 = 6.8 nM T51408 C6D5IZ 46881618 EC50 = 174 nM T51408 CTC02J 46881650 EC50 = 74 nM T51408 CN9TK8 46881651 EC50 = 86 nM T51408 CWZ4H5 46881652 EC50 = 8 nM T51408 CZQ6C8 46881653 EC50 = 171 nM T51408 CD27OS 46881698 EC50 = 64 nM T51408 CGP45C 46881699 EC50 = 19 nM T51408 C7BPN3 46881700 EC50 = 19 nM T51408 CMR6C9 46881701 EC50 = 16 nM T51408 C8QS6V 46881750 EC50 = 283 nM T51408 C8XST7 46881751 EC50 = 2647 nM T51408 CW60AO 46881752 EC50 > 10 nM T51408 CFIE98 46881753 EC50 = 454 nM T51408 C4EOF8 46881796 EC50 = 261 nM T51408 C9HO2J 46881797 EC50 = 580 nM T51408 CX8ZS6 46881798 EC50 = 218 nM T51408 C9OE3N 46881799 EC50 = 241 nM T51408 CV75XD 46881838 EC50 = 123 nM T51408 CVR9M2 46881839 EC50 = 498 nM T51408 C4D1XF 46881840 EC50 = 10 nM T51408 CK0N6A 46881869 EC50 = 3768 nM T51408 C9CUP4 46881870 EC50 = 1404 nM T51408 C53CIB 46881871 EC50 = 1.9 nM T51408 CGZ7K5 46881872 EC50 = 978 nM T51408 CHJ9D1 46881899 EC50 = 179 nM T51408 C4D7PW 46881900 EC50 = 184 nM T51408 CI7Q6U 46881901 EC50 = 187 nM T51408 CTX8N0 46881902 EC50 = 67 nM T51408 CR1H5N 46881935 EC50 = 76.2 nM T51408 CQ87KZ 46881936 EC50 = 21 nM T51408 CKDO83 46881937 EC50 = 36 nM T51408 C7W1LE 46881938 EC50 = 42 nM T51408 CXDJ80 46881980 EC50 = 86 nM T51408 CP5O9V 46881981 EC50 = 24 nM T51408 C4N0KV 46881982 EC50 = 32 nM T51408 C50CFL 46881983 EC50 = 35 nM T51408 C50GNW 46882028 EC50 = 47 nM T51408 CBC6Z5 46882029 EC50 = 6.9 nM T51408 C2Y3DO 46882030 EC50 = 10 nM T51408 CWG7Z8 46882031 EC50 = 37 nM T51408 CWI86A 46882084 EC50 = 105 nM T51408 CMC4E5 46882804 IC50 = 5200 nM T51408 CBN3V6 46889642 Ki = 8500 nM T51408 CG72PB 46889643 Ki = 1000 nM T51408 C8S4LM 46889670 Ki = 225 nM T51408 CEF90S 46889699 Ki = 2340 nM T51408 CH4Z0F 46889700 Ki = 3820 nM T51408 C8K6HX 46889701 Ki = 2200 nM T51408 CAO57K 46889727 Ki = 1510 nM T51408 CTP3E7 46889728 Ki = 698 nM T51408 CW9LS6 46889729 Ki = 3400 nM T51408 C7RI4K 46889730 Ki = 1480 nM T51408 C4ISX8 46889767 Ki = 11000 nM T51408 C3ZY5J 46889768 Ki = 2900 nM T51408 C3F4IQ 46889769 Ki = 6225 nM T51408 C1P5WV 46889770 Ki = 1060 nM T51408 C02HNI 46889771 EC50 = 234 nM T51408 C4D5FH 46889772 Ki = 410 nM T51408 CKIM07 46889809 Ki = 98 nM T51408 C6CY1S 46889810 Ki = 230 nM T51408 C26WTA 46889811 Ki = 455 nM T51408 C2GC4K 46889812 Ki = 72 nM T51408 C9P4TD 46889852 Ki = 230 nM T51408 C1YVO4 46889853 Ki = 9180 nM T51408 CFY40T 46889854 Ki = 250 nM T51408 CK8V2H 49800025 EC50 = 25.12 nM T51408 CV5G1H 49861320 EC50 = 520 nM T51408 C2RY0J 50878551 Ki > 10000 nM T51408 C1W6TV 50898777 Ki > 10000 nM T51408 CXMZ73 50898778 Ki > 10000 nM T51408 CLY9W1 50994950 EC50 = 63 nM T51408 C2CH1R 50995330 EC50 = 24 nM T51408 CE4KP1 51050257 Ki > 10000 nM T51408 CYR21W 51346867 EC50 = 4.1 nM T51408 CJ9L0W 51347282 EC50 = 43 nM T51408 C4Z2FY 51347436 EC50 = 0.64 nM T51408 CQG7X2 51349173 EC50 = 18 nM T51408 C1F0DX 52941476 Ki = 63 nM T51408 C6VLH4 52941547 EC50 = 150 nM T51408 CZMS46 52941603 EC50 = 55 nM T51408 C6J0HT 52941935 EC50 = 150 nM T51408 CZ1G5T 52942807 EC50 = 150 nM T51408 C83BMV 52943362 EC50 = 4.7 nM T51408 C3B2OF 52943383 Ki = 59 nM T51408 C3EO6J 52943730 Ki = 770 nM T51408 C61ZLX 52943770 EC50 = 1.2 nM T51408 CE13YX 52943919 EC50 = 79 nM T51408 C5TW1N 52943932 EC50 = 35 nM T51408 CVE5Q9 52943968 Ki = 37 nM T51408 C69LKY 52943969 Ki = 85 nM T51408 C1AXC6 52944896 EC50 = 150 nM T51408 CP6U9S 52944986 EC50 = 8.3 nM T51408 C0TWA8 52946357 EC50 = 1.7 nM T51408 CFX1D5 52946430 Ki = 331 nM T51408 CI2PT6 52946537 EC50 = 2.8 nM T51408 C7ULQ8 52947060 Ki = 90 nM T51408 CB5ZY1 52947431 Ki = 3300 nM T51408 CHK30N 52947443 Ki = 17 nM T51408 CQR7T0 52947487 EC50 = 150 nM T51408 CD7EW1 52947562 EC50 = 15 nM T51408 C5ED6I 52947654 EC50 = 150 nM T51408 CED37H 52948056 EC50 = 10 nM T51408 C5BEO2 52948572 EC50 = 150 nM T51408 CN0F9Z 52948612 EC50 = 2410 nM T51408 CBXN18 52948613 Ki = 370 nM T51408 C04PTF 52948728 EC50 = 24 nM T51408 C6E9TK 52948792 Ki = 107 nM T51408 CU1R7B 52948805 Ki = 64 nM T51408 CI7S6O 52949488 EC50 = 2.5 nM T51408 CMX86D 52949489 EC50 = 21 nM T51408 CD68KM 52949862 Ki = 8000 nM T51408 C9VYT6 52949934 EC50 = 7.1 nM T51408 C79TFR 52950121 EC50 = 150 nM T51408 C57DOH 53318280 EC50 = 11 nM T51408 CJAH78 53319639 EC50 = 1307 nM T51408 CA45EM 53326195 EC50 = 15 nM T51408 C9SDC2 53326196 EC50 = 2030 nM T51408 CM5WF2 53326197 EC50 = 8.3 nM T51408 C3EAT2 53326839 EC50 = 81 nM T51408 CLN6B9 53357711 EC50 = 100 nM T51408 CL7US4 53357712 EC50 = 63.1 nM T51408 CRGV73 56597179 EC50 = 10000 nM T51408 CB8O9W 56598831 EC50 = 10000 nM T51408 CQKF90 56598832 EC50 = 10000 nM T51408 CR6PU5 56598833 EC50 = 10000 nM T51408 CRO1Y2 56598967 EC50 = 10000 nM T51408 C43AZK 56658246 EC50 = 398.11 nM T51408 CCAE43 56658405 EC50 = 12.59 nM T51408 CMWZ90 56658407 EC50 = 15.85 nM T51408 CPE84D 56665368 EC50 = 158.49 nM T51408 CEU7B9 56668796 EC50 = 12.59 nM T51408 C9CRA4 56672269 EC50 = 31.62 nM T51408 CM3YO8 56672271 EC50 = 100 nM T51408 CLB1V0 56675663 EC50 = 25.12 nM T51408 CE5DQ6 56678849 EC50 = 25.12 nM T51408 CT2E1Z 56678973 EC50 = 2.512 nM T51408 C6T7YR 56943485 EC50 = 50.12 nM T51408 C7DEO8 56943515 EC50 = 39.81 nM T51408 CZF4B5 56943517 EC50 = 31.62 nM T51408 CJ81YS 56943518 EC50 = 39.81 nM T51408 C5M0CT 56943545 EC50 = 39.81 nM T51408 CMUQ15 56943546 EC50 = 39.81 nM T51408 C1TC7Q 56963799 Ki > 10000 nM T51408 C5BSH0 66653268 EC50 = 10000 nM T51408 CS2K0M 66796015 EC50 = 39.81 nM T51408 C3ARI1 67972106 EC50 = 3.3 nM T51408 CXJ68U 67972107 EC50 = 1.7 nM T51408 CB05ID 67972431 EC50 = 20 nM T51408 C7WL6M 68155065 EC50 = 309 nM T51408 CPX1H7 69119729 EC50 = 398.11 nM T51408 CV57BY 69119831 EC50 = 316.23 nM T51408 C86CXO 69119890 EC50 = 251.19 nM T51408 C4H3LN 69120058 EC50 = 398.11 nM T51408 CNVH59 69442961 EC50 = 1995.26 nM T51408 CKWP40 69447283 EC50 = 2511.89 nM T51408 CW9KA8 69655138 EC50 = 260 nM T51408 CBDL19 70792359 EC50 = 3.7 nM T51408 C6T0KD 71459884 Ki = 14100 nM T51408 CC65OA 73213195 Ki > 10000 nM T51408 CW83DK 73213196 Ki > 10000 nM T51408 C7TM8S 73349644 EC50 = 270 nM T51408 C74QNU 73352659 EC50 = 400 nM T51408 CG0Z2D 73357212 EC50 = 280 nM T51408 CVY13Q 76314766 EC50 = 16.7 nM T51408 C5ZDK4 76315637 EC50 = 1.2 nM T51408 CFZU52 76315638 EC50 = 0.54 nM T51408 C0X7CQ 76315639 EC50 = 160 nM T51408 CGZ5C4 76315640 EC50 = 4.4 nM T51408 C67YUD 76318362 EC50 = 12.4 nM T51408 C1M4TQ 76318363 EC50 = 76.7 nM T51408 CCUG71 76318364 EC50 = 0.83 nM T51408 C9PM0U 76319327 EC50 = 1.3 nM T51408 CR05PL 76322043 EC50 = 1.36 nM T51408 CQ3CW1 76322044 EC50 = 1.15 nM T51408 CFU26T 76322045 EC50 = 186 nM T51408 CTD25H 76322046 EC50 = 44.2 nM T51408 C61AMT 76322047 EC50 = 0.21 nM T51408 CI8XA7 76322965 EC50 = 1 nM T51408 CQI0H5 76325667 EC50 = 1.95 nM T51408 C6R4BP 76325668 EC50 = 13.6 nM T51408 CB71EI 76325669 EC50 = 0.88 nM T51408 C03YTR 76329059 EC50 = 3981.07 nM T51408 CRW8C5 76329232 EC50 = 0.48 nM T51408 C5SKR4 76332892 EC50 = 8.78 nM T51408 CMR86G 76332893 EC50 = 1.86 nM T51408 CTVI40 76332894 EC50 = 0.04 nM T51408 CL7TN0 76332895 EC50 = 0.13 nM T51408 C8PGV1 76333795 EC50 = 0.47 nM T51408 CQ47BW 76336499 EC50 = 1.6 nM T51408 C92WBQ 76336500 EC50 = 0.15 nM T51408 C8KBZ1 76336501 EC50 = 0.15 nM T51408 CQM69X 76336502 EC50 = 0.37 nM T51408 CNXH73 90645344 EC50 = 6.31 nM T51408 C9W1FB 90645345 EC50 = 12.59 nM T51408 CR7OT8 90645346 EC50 = 12.59 nM T51408 C9A5KY 90645347 EC50 = 7.943 nM T51408 CQNL51 118725301 EC50 = 10000 nM T51408 CUK7B0 122184771 EC50 = 71 nM T51408 CX7U6O 122184772 EC50 = 43 nM T51408 CNT76C 122184833 EC50 = 338 nM T51408 C8C2KW 122184834 EC50 > 10000 nM T51408 CGNH50 122184835 EC50 = 111 nM T51408 C1CJQ0 122188571 Ki = 1440 nM T51408 C4D9QY 127026491 EC50 = 2.6 nM T51408 C7L1DB 127037832 EC50 = 2.1 nM T51408 CG84RM 127041558 EC50 = 1.9 nM T51408 CS20QX 127041559 EC50 = 9.7 nM T51408 CN2T3I 127041869 EC50 = 0.49 nM T51408 C2BE3M 127041870 EC50 = 3.1 nM T51408 C31SDE 127042181 EC50 = 5.4 nM T51408 C6UOA4 127042536 EC50 = 3.7 nM T51408 CD0FI8 135995975 EC50 = 90 nM T51408 CD96BP 135995976 EC50 = 34 nM T51408 CU7Q8F 135995977 EC50 = 80 nM T51408 C29TCN 135995978 EC50 = 10 nM T51408 C2QCA5 137631487 EC50 = 5.1 nM T51408 C8HPN4 137634334 EC50 = 1.6 nM T51408 CVER86 137640335 EC50 = 18 nM T51408 C70XZQ 137643636 EC50 = 2.9 nM T51408 CL06NY 137648464 EC50 = 1.9 nM T51408 CUFO39 137649223 EC50 = 0.32 nM T51408 C65XKJ 137653127 EC50 = 2.5 nM T51408 C3LG7W 137655838 EC50 = 5.2 nM T51408 CN2UE9 137656598 EC50 = 1.5 nM T51408 CB8C3F 137657762 EC50 = 6.5 nM T51408 CT5CX0 145973771 Ki = 2360 nM T51408 C72IAC 145980824 EC50 > 10000 nM T51408 CNA4W1 145982519 EC50 = 4.623 nM T51408 CBNQ70 145982607 EC50 = 8.683 nM T51408 C6MWR1 145982668 EC50 = 7.699 nM T51408 CMHJ54 145983042 EC50 = 10.45 nM T51408 CSB96G 145983164 EC50 = 1.422 nM T51408 CFBS76 145983266 EC50 = 3.412 nM T51408 CZ60KX 145983355 EC50 = 11.14 nM T51408 CKX16A 145983603 EC50 = 1.029 nM T51408 C82XTN 145983617 EC50 = 2.616 nM T51408 CH3LJ5 145983629 EC50 = 2.491 nM T51408 COZ4J2 145983711 EC50 = 4.699 nM T51408 CN0D9C 145983745 EC50 = 1.493 nM T51408 C9C6RI 145983829 EC50 = 2.082 nM T51408 CF0J8G 145983886 EC50 = 8.435 nM T51408 CLWN42 145984040 EC50 = 1.782 nM T51408 C9DX1E 145984042 EC50 = 4.584 nM T51408 CD3J9G 145984044 EC50 = 1.653 nM T51408 CT4BM0 145984324 EC50 = 55.45 nM T51408 CCA7F4 145984563 EC50 = 2.927 nM T51408 CE5PC2 145984584 EC50 = 0.5117 nM T51408 C8UP3K 145984667 EC50 = 3.575 nM T51408 C82AHK 145984792 EC50 = 7.805 nM T51408 CH7MX0 145985242 EC50 = 1.089 nM T51408 CA67ZV 145985368 EC50 = 2.894 nM T51408 CRS15X 145985509 EC50 = 2.153 nM T51408 C1ZWI5 145986105 EC50 = 1.424 nM T51408 CK1C0A 145989075 EC50 > 10000 nM T51408 C4GV8Q 145990586 IC50 = 240 nM T51408 C0SH3Y 145991661 EC50 > 10000 nM T51408 CV7U8T 145994130 EC50 > 10000 nM T51408 C6P3SR 153287553 Ki > 10000 nM T51408 CV9G7Z 153287572 Ki > 10000 nM T51408 CO85KL 153287574 Ki = 1000 nM T51408 CUSA24 155519891 Ki > 10000 nM T51408 CV83SG 155534733 Ki = 1420 nM T51408 CB79ZW 155536080 Ki > 10000 nM T51408 CP9TR0 10324985 Ki > 10000 nM T51408 CF40LD 44349237 EC50 = 120 nM T51408 CTNO31 44349323 EC50 = 300 nM T51408 C91AXH 44349356 EC50 = 140 nM T51408 C9JZ7V 44349357 EC50 = 180 nM T51408 C5TWZ0 44349367 EC50 = 35 nM T51408 CE2XL3 44349378 EC50 = 22 nM T51408 C5ELB7 44349379 EC50 = 10 nM T51408 D01OIK 155774 EC50 = 100000 nM T51408 D02DKX 5311116 EC50 = 10000 nM T51408 D03BZW 2687 EC50 = 2000 nM T51408 D03VHK 10028830 EC50 = 11.91 nM T51408 D04HXF 4080436 Ki = 1770 nM T51408 D0A4FU 2769774 Ki = 4960 nM T51408 D0H3WJ 44435193 Ki = 2500 nM T51408 D0L5MW 181743 Ki > 10000 nM T51408 D0YZ3E 44435200 Ki = 1700 nM T64205 D09ZCV 73333953 IC50 = 10900 nM T64205 D0EX9O 68075823 IC50 = 5800 nM T64205 D0XQ3F 9870708 IC50 = 42000 nM T64205 D0Y0OQ 24767791 Ki > 25000 nM T64205 CZ25OS 8514 IC50 = 9100 nM T64205 C8U1AQ 658668 IC50 > 50000 nM T64205 CV01HZ 665421 IC50 > 50000 nM T64205 C5C9AV 665426 IC50 > 50000 nM T64205 CX17KE 665524 IC50 > 50000 nM T64205 CYR0A9 665706 IC50 > 50000 nM T64205 C07LUC 665766 IC50 > 50000 nM T64205 CG69BA 665910 IC50 > 50000 nM T64205 CE6JB5 1383290 IC50 > 50000 nM T64205 CSQ26L 1400670 IC50 > 50000 nM T64205 CZJN05 1409627 IC50 = 40600 nM T64205 CK27XL 3592521 IC50 > 50000 nM T64205 CLE8J0 4378002 IC50 > 50000 nM T64205 CL1A9Z 4744091 IC50 > 50000 nM T64205 CORG34 9566174 IC50 = 130000 nM T64205 C7BG3Z 10895852 IC50 = 10000 nM T64205 CN89IB 16730520 IC50 = 560000 nM T64205 CP28EL 24768184 IC50 = 210000 nM T64205 CI28CQ 24768185 IC50 = 605000 nM T64205 C37AZQ 24768186 IC50 = 380000 nM T64205 CB5RJ6 24768187 IC50 = 760000 nM T64205 C2B5CI 24768188 IC50 = 250000 nM T64205 CXBZ69 24768189 IC50 = 402000 nM T64205 CF15NC 56663448 Ki = 9700 nM T64205 CZI54O 56673821 Ki = 22000 nM T64205 CO7R8N 56680467 Ki = 8800 nM T64205 C0HSI2 56847442 Ki > 25000 nM T64205 CSL3N8 68075861 Ki = 3200 nM T64205 CU61YT 68075994 Ki > 25000 nM T64205 CAYX80 68076759 Ki > 25000 nM T64205 CT2G3X 70681428 Ki = 9500 nM T64205 C1VM0Q 70681429 Ki = 27800 nM T64205 CCNS57 71311907 IC50 = 33200 nM T64205 C4A0EX 90643506 IC50 = 11800 nM T64205 C2BR1Z 90643507 IC50 = 50700 nM T64205 CD4IR5 90665637 IC50 = 7200 nM T64205 C34BNA 118714785 IC50 > 30000 nM T64205 CSMF46 118714786 IC50 > 30000 nM T64205 C5MXD3 118714787 IC50 > 30000 nM T64205 C1L6DR 118714788 IC50 > 30000 nM T64205 CXAK53 118714789 IC50 > 30000 nM T64205 CO4ZX1 118714790 IC50 > 30000 nM T64205 C80IVZ 118714791 IC50 > 30000 nM T64205 C1Z8UW 118714792 IC50 > 30000 nM T64205 CS4Y6R 118714793 IC50 > 30000 nM T64205 CGO49H 121485603 IC50 > 50000 nM T64205 CQD86F 122417980 IC50 > 50000 nM T64205 CWP4Y3 127043537 IC50 > 50000 nM T64205 CD4PS6 127043538 IC50 > 50000 nM T64205 C62JRB 127043708 IC50 > 50000 nM T64205 CRMT13 127043884 IC50 > 50000 nM T64205 CVQR69 127043885 IC50 > 50000 nM T64205 CWT75I 127043886 IC50 > 50000 nM T64205 CBPX56 127043998 IC50 = 45900 nM T64205 C5J8LF 127044001 IC50 > 50000 nM T64205 CDO20J 127044052 IC50 > 50000 nM T64205 CN27VG 127044282 IC50 > 50000 nM T64205 CNJ8A1 127044345 IC50 > 50000 nM T64205 CWM68F 127044476 IC50 > 50000 nM T64205 C65KPY 127044624 IC50 > 30000 nM T64205 CA6WV5 127044625 IC50 = 29500 nM T64205 CIXY97 127044626 IC50 > 50000 nM T64205 C7MIB0 127044627 IC50 > 50000 nM T64205 CP0KI6 127044628 IC50 > 50000 nM T64205 CJ5SF0 127044631 IC50 > 50000 nM T64205 C4PV9O 127044955 IC50 = 15000 nM T64205 CF3IT2 127045104 IC50 > 30000 nM T64205 CKRU47 134135130 IC50 = 7000 nM T64205 C0XZ6L 134145005 IC50 = 2000 nM T64205 CKS5Y9 134148443 IC50 > 50000 nM T64205 C0IVR3 134151103 IC50 = 2000 nM T64205 C1QXI7 135402276 IC50 > 50000 nM T64205 CBN8M7 135449231 IC50 = 12100 nM T64205 CJ58AO 135463175 IC50 > 50000 nM T64205 D0D9AA 6093161 IC50 = 7900 nM T98022 D05WSP 11241908 Ki = 10 nM T98022 D0F7FX 87609775 IC50 = 400 nM T98022 CMU34O 9813856 IC50 = 36 nM T98022 CRI52O 9816170 Ki = 46 nM T98022 CC60TU 9834324 IC50 = 26000 nM T98022 CK2O8T 9834556 IC50 = 15000 nM T98022 C40BDL 9834739 IC50 = 100 nM T98022 C7PMN6 9834740 IC50 = 5800 nM T98022 CF5A3T 9837547 IC50 = 35 nM T98022 CDJW45 9855661 IC50 = 6800 nM T98022 CYW97I 9856625 IC50 = 5300 nM T98022 CQ6HP2 9857137 IC50 = 6 nM T98022 CV71OD 9877989 IC50 = 12000 nM T98022 CLGB62 9888695 IC50 = 5.5 nM T98022 CWH57U 9899367 IC50 > 50000 nM T98022 C0J5IB 9899633 IC50 = 1500 nM T98022 CV6F0Y 9900049 IC50 = 24 nM T98022 CKQP09 9920759 IC50 = 4700 nM T98022 CJ53NX 9921072 IC50 > 20000 nM T98022 CHI95J 9926432 IC50 = 4 nM T98022 C9WT3L 9942902 IC50 = 50 nM T98022 CM1A0D 9943447 IC50 = 52 nM T98022 C4ZBI0 9964544 IC50 > 20000 nM T98022 CY8UR1 9964714 IC50 = 7000 nM T98022 C93GRP 9964715 IC50 > 20000 nM T98022 CW28EQ 9966944 IC50 = 21 nM T98022 C39EUV 10149451 Ki = 7.5 nM T98022 CX4KD6 10192710 IC50 = 1070 nM T98022 CBP24H 10198140 IC50 = 139 nM T98022 C5RFA9 10214532 IC50 = 45 nM T98022 C68FIU 10214568 IC50 = 3 nM T98022 C5YRO9 10236323 IC50 = 11 nM T98022 CK05UJ 10308002 IC50 = 5300 nM T98022 C73LOJ 10308062 IC50 = 7350 nM T98022 C5G7KU 10308323 Ki = 5.8 nM T98022 CVK4L6 10418061 IC50 = 1.5 nM T98022 C6FQ0R 10465893 IC50 > 100000 nM T98022 CXT3L1 11149158 Ki = 84 nM T98022 CZOS28 11172834 Ki = 100 nM T98022 C8OFL4 11241046 Ki = 344 nM T98022 C84FJY 11334286 Ki = 70 nM T98022 CT7IR8 12110710 IC50 = 1.9 nM T98022 C41JOB 15342746 IC50 = 400 nM T98022 C3U6FC 15974385 Ki > 700 nM T98022 CAYN20 21303381 Ki = 407 nM T98022 C2ZV4R 22289844 Ki = 65 nM T98022 C9H4OA 22319346 Ki = 140 nM T98022 C75JHY 22319377 IC50 = 620 nM T98022 CW71PB 23730599 Ki = 160 nM T98022 C24ZKE 23730600 Ki = 140 nM T98022 CE1G2T 23730827 Ki = 235 nM T98022 C9K4XA 23730828 Ki = 250 nM T98022 CI32BD 23730940 Ki = 430 nM T98022 C1ATY0 23730941 Ki = 269 nM T98022 CO7WS2 23730942 Ki = 124 nM T98022 CF4TP1 23730943 Ki = 111 nM T98022 C0K3MY 25159540 IC50 = 850 nM T98022 CN4R0T 25159662 IC50 = 170 nM T98022 C0Z8WA 25159800 IC50 = 59000 nM T98022 C7UMS0 25160056 IC50 = 1200 nM T98022 C4Q6MH 25160058 IC50 = 39 nM T98022 C3M1VF 25160194 IC50 = 110 nM T98022 CQ9T1K 25160196 IC50 = 900 nM T98022 C8HK2A 25160206 IC50 = 5700 nM T98022 C7W3VM 25160334 IC50 = 190 nM T98022 CL3T4D 25160336 IC50 = 120 nM T98022 CBHS65 25160458 IC50 = 690 nM T98022 C05QKN 44308084 IC50 = 380 nM T98022 CR1H5M 44308085 IC50 > 20000 nM T98022 CD05IM 44308178 IC50 = 13000 nM T98022 CS5OI1 44308185 IC50 > 20000 nM T98022 C1HCY9 44308186 IC50 = 270 nM T98022 CHQF08 44308224 IC50 > 20000 nM T98022 CNCO42 44308235 IC50 = 3300 nM T98022 CD7IK4 44308237 IC50 = 1 nM T98022 C9IPN5 44308238 IC50 = 100 nM T98022 C5ZWR2 44308262 IC50 = 6700 nM T98022 CR2MV9 44308268 IC50 = 67000 nM T98022 CBR39F 44308352 IC50 = 2 nM T98022 CH27SZ 44308370 IC50 = 12 nM T98022 C5LY4T 44308385 IC50 = 23 nM T98022 CG31EH 44308398 IC50 > 20000 nM T98022 CBDE72 44308420 IC50 > 20000 nM T98022 CN3ZR7 44308432 IC50 > 20000 nM T98022 C6SV1C 44387258 IC50 = 1.5 nM T98022 CIP46H 44436064 Ki = 17000 nM T98022 C6CT7P 44440388 IC50 = 905 nM T98022 C28NTH 44440390 IC50 = 92 nM T98022 CZY78Q 46225030 Ki = 6.7 nM T98022 CEQ39A 46225031 Ki = 5.7 nM T98022 CITR87 46225064 Ki = 8.2 nM T98022 CQH24P 46225065 Ki = 15 nM T98022 CB3ZI1 46225066 Ki > 1000 nM T98022 CHNY62 59187273 IC50 = 230 nM T98022 C4LY2E 59187280 IC50 = 670 nM T98022 C03RKH 59187282 IC50 = 31 nM T98022 CR06PG 59187284 IC50 = 69 nM T98022 CQXH69 59187288 IC50 = 490 nM T98022 C5S2PW 59187291 IC50 = 220 nM T98022 CMI2O3 59187303 IC50 = 1400 nM T98022 CN6V2H 59187309 IC50 = 400 nM T98022 CQ0NR9 59187313 IC50 = 71 nM T98022 C57VUW 59187317 IC50 = 200 nM T98022 CJ26WC 59187318 IC50 = 1100 nM T98022 C2I0US 59187319 IC50 = 360 nM T98022 C89TSD 59187321 IC50 = 1100 nM T98022 CQ90KX 59187323 IC50 = 6700 nM T98022 C29TQV 59187327 IC50 = 1100 nM T98022 C7Y3EM 59187328 IC50 = 110 nM T98022 C4F0EO 59187329 IC50 = 1700 nM T98022 CLWJ12 59187334 IC50 = 130 nM T98022 CXQ2D4 59187337 IC50 = 130 nM T98022 CR2M0O 59187340 IC50 = 49 nM T98022 C3S4DN 59187343 IC50 = 2100 nM T98022 CF9O8P 59187344 IC50 = 170 nM T98022 C5JU2Z 59187346 IC50 = 390 nM T98022 C6KT3I 59187348 IC50 = 1700 nM T98022 CW42HM 59187351 IC50 = 2300 nM T98022 CUW75B 59187356 IC50 = 19 nM T98022 C8E1KM 59187365 IC50 = 7100 nM T98022 CZ6HS9 59187366 IC50 = 1700 nM T98022 CD3UC7 59187369 IC50 = 170 nM T98022 C59TNF 66563223 IC50 = 30 nM T98022 C7UY0I 66563225 IC50 = 1.1 nM T98022 CSX85Y 66563227 IC50 = 1600 nM T98022 CK3OI1 66563229 IC50 = 5.3 nM T98022 CO1AD9 66563231 IC50 = 180000 nM T98022 CX8WC6 66563346 IC50 = 2600 nM T98022 C2NZM7 66563348 IC50 = 2 nM T98022 CT0AE1 66563350 IC50 = 200 nM T98022 C5RSJ8 66563352 IC50 = 0.025 nM T98022 C38FZA 71451543 IC50 = 62000 nM T98022 CUCW23 71451544 IC50 = 3800 nM T98022 CC39TP 71455084 IC50 = 310000 nM T98022 CDN5R9 71456891 IC50 = 34 nM T98022 CM24UO 76871913 IC50 = 76 nM T98022 C5Y9UI 87901223 IC50 = 15000 nM T98022 CBX7L2 90655303 IC50 < 41 nM T98022 CHZ2M5 90655305 IC50 = 80 nM T98022 CPH9G2 90655306 IC50 = 106 nM T98022 C9Z3YM 90655307 IC50 = 124 nM T98022 CI31SH 90655308 IC50 = 585 nM T98022 CIC01B 90655309 IC50 = 2270 nM T98022 CN49KI 90655310 IC50 = 66 nM T98022 C5MBY1 90655311 IC50 < 41 nM T98022 C0NF1Z 91799224 IC50 = 1500 nM T98022 C0H8AW 122177723 IC50 = 3 nM T98022 CFZ05M 122177724 IC50 = 15 nM T98022 C6MTR2 122177725 IC50 = 57 nM T98022 CXY64B 122177726 IC50 = 460 nM T98022 C7DS2R 122177727 IC50 = 1000 nM T98022 C2ZG4X 122177728 IC50 = 3700 nM T98022 CJY8F2 122177729 IC50 = 6100 nM T98022 CF48KT 122177730 IC50 = 15 nM T98022 CCS01U 122177731 IC50 = 7 nM T98022 C5AZW6 122177732 IC50 = 9 nM T98022 CE46VD 122177733 IC50 = 4 nM T98022 CIL19A 122177734 IC50 = 18 nM T98022 CJ6B2T 122177735 IC50 = 38 nM T98022 CS3LA9 122177736 IC50 = 4 nM T98022 CAJ26V 122177737 IC50 = 4 nM T98022 CKM2V8 122177738 IC50 = 100 nM T98022 CG1CR4 122177739 IC50 = 1 nM T98022 C1SX5C 122177740 IC50 = 250 nM T98022 CAE8Q5 122177741 IC50 = 750 nM T98022 CQ2B5S 122177742 IC50 = 570 nM T98022 CQ0LM1 122177743 IC50 = 54000 nM T98022 CXU38V 122197590 IC50 = 12 nM T98022 C7WD2Q 134133082 IC50 > 30000 nM T98022 C45ZGT 134133657 IC50 > 30000 nM T98022 CPN13Y 134136702 IC50 = 75000 nM T98022 C0JL8S 134136841 IC50 > 30000 nM T98022 CU87CW 134137231 IC50 = 1700 nM T98022 C0RE6H 134138207 IC50 = 24000 nM T98022 C3QVD6 134140975 IC50 > 30000 nM T98022 C8QHO4 134142117 IC50 = 3 nM T98022 CO3XS7 134142683 IC50 > 30000 nM T98022 C46VIY 134142802 IC50 = 880 nM T98022 C4YPT3 134142983 IC50 = 26 nM T98022 C8XDV4 134144273 IC50 = 1500 nM T98022 CFV04E 134144803 IC50 = 10000 nM T98022 CSLZ67 134144998 IC50 = 44000 nM T98022 CCG3E8 134146335 IC50 > 30000 nM T98022 C2HN0T 134146423 IC50 > 30000 nM T98022 CYK8C3 134147307 IC50 = 38 nM T98022 CSM4H3 134148649 IC50 = 420 nM T98022 C12FRQ 134149241 IC50 > 30000 nM T98022 CIV3Q1 134151262 IC50 = 4400 nM T98022 C4HC8J 134151680 IC50 = 330 nM T98022 C4MZ8F 134153015 IC50 > 30000 nM T98022 CB9A4L 134154540 IC50 = 47000 nM T98022 C1GF8Q 134155782 IC50 = 81 nM T98022 CLM28S 134157143 IC50 = 6400 nM T98022 C7AFS1 134157353 IC50 = 51 nM T98022 CB3W0T 145961938 IC50 = 1.5 nM T98022 D00DXB 10214441 IC50 = 68 nM T98022 D00GOD 10035600 IC50 = 590 nM T98022 D06LNX 3858 IC50 = 1600 nM T98022 D06TJC 10192614 IC50 = 37 nM T98022 D0JD9E 194328 Ki = 4 nM T98022 D0O3QJ 10286113 Ki = 3.5 nM T98022 D0R2PW 10214451 IC50 = 785 nM T98022 D0R7PE 20384315 Ki = 300 nM T91940 D06NVJ 936 IC50 = 46600 nM T91940 D0E7PQ 5311 IC50 > 100000 nM T91940 D0Y3KG 3121 IC50 > 100000 nM T91940 D0B7CH 4775 IC50 > 100000 nM T91940 D0H2UB 5361 IC50 = 22000 nM T91940 D04JZE 3246390 IC50 = 42500 nM T91940 C85KQB 2202 IC50 = 100 nM T91940 C0J1SW 694859 IC50 = 39400 nM T91940 CBD84H 698853 IC50 = 12600 nM T91940 C3VBZ9 1095092 IC50 = 3600 nM T91940 C6YS9Z 1103548 IC50 = 12400 nM T91940 CE4KD6 1142691 IC50 = 16600 nM T91940 CB92ZQ 1372991 IC50 = 6200 nM T91940 CX8WT2 2248572 IC50 = 25200 nM T91940 CDWU19 2827646 IC50 = 48900 nM T91940 C94ELI 3610426 IC50 = 30000 nM T91940 CQ5NA2 7333748 IC50 = 67300 nM T91940 C6L5KB 45168044 IC50 > 100000 nM T91940 CC7T2A 56674921 IC50 = 19500 nM T91940 CUSF78 57327892 IC50 = 5000 nM T91940 C8CLX3 71452171 IC50 = 17800 nM T91940 C73LSH 71453984 IC50 = 12900 nM T91940 C1O0HF 71459392 IC50 = 22400 nM T91940 CQM08D 121231415 IC50 > 200000 nM T91940 C5Y9AJ 122184880 IC50 > 100000 nM T91940 CR86MS 122184881 IC50 = 5000 nM T91940 CY9D7A 122184882 IC50 > 100000 nM T91940 C0H4GO 122184884 IC50 > 100000 nM T91940 CML8G1 122186876 IC50 = 2000000 nM T91940 CH2BJ7 124156324 IC50 > 200000 nM T91940 CZDJ49 124156728 IC50 > 200000 nM T91940 CU4IC8 126843233 IC50 > 200000 nM T91940 CYAK84 134141382 IC50 > 200000 nM T91940 C7B5KW 134142322 IC50 > 400000 nM T91940 CC4Z9Q 134143263 IC50 > 6000000 nM T91940 C53ATF 134148970 IC50 > 2000000 nM T91940 CRON29 134150759 IC50 > 300000 nM T91940 C9YPF1 134820907 IC50 > 100000 nM T91940 CB53GJ 135443018 IC50 = 46500 nM T91940 C4KDT9 135457159 IC50 = 27000 nM T91940 CW50RD 135469837 IC50 = 55900 nM T91940 C91HDU 137631681 IC50 = 46.1 nM T91940 C0TC5F 137632075 IC50 = 2673 nM T91940 C8X4NQ 137632345 Ki = 263 nM T91940 CPJ5T8 137632865 IC50 = 714.5 nM T91940 C01GMZ 137632891 IC50 = 893.3 nM T91940 CB1L5T 137633463 Ki = 3.5 nM T91940 C6N2UG 137634133 IC50 = 1606.9 nM T91940 C01LYF 137634283 Ki = 3.5 nM T91940 C13CJM 137634356 IC50 = 2060.6 nM T91940 C9QJ6R 137635476 IC50 = 2202.7 nM T91940 CXB14F 137636901 IC50 = 12502.6 nM T91940 CR4N5F 137637122 IC50 = 207 nM T91940 CVK0C5 137637617 Ki = 13.6 nM T91940 CUJE57 137638306 IC50 = 1614.4 nM T91940 CCX69V 137638847 IC50 > 40000 nM T91940 C2FTJ4 137639138 IC50 = 5600 nM T91940 C1DE6B 137639267 IC50 = 647.1 nM T91940 C0IPW8 137639647 IC50 = 1181 nM T91940 CF74SI 137639873 IC50 = 1111.7 nM T91940 C8A1KL 137639921 IC50 = 72560 nM T91940 CK28IL 137640497 Ki = 3.5 nM T91940 C9Z5UY 137640785 IC50 = 779.8 nM T91940 CGD68K 137640803 IC50 = 325.8 nM T91940 CU20QE 137640903 IC50 = 157200 nM T91940 C59BKE 137641229 IC50 = 1047.1 nM T91940 C3TB9Y 137641253 IC50 = 1124.6 nM T91940 CBP1U5 137642419 Ki = 83.2 nM T91940 C6MWL3 137642629 Ki = 7 nM T91940 CUB63V 137643467 IC50 > 14000 nM T91940 C13VQS 137643947 IC50 = 1977 nM T91940 CO1FY4 137644287 IC50 = 7500 nM T91940 CORN56 137644685 IC50 = 1235.9 nM T91940 C9Q2ZE 137644712 IC50 = 2741.6 nM T91940 CL52GA 137644801 IC50 = 335.7 nM T91940 CRO0W9 137645261 IC50 = 4027.2 nM T91940 C9KYV4 137645360 IC50 = 59 nM T91940 CAH95W 137646179 IC50 = 1383.6 nM T91940 CTR34G 137647267 IC50 = 1129.8 nM T91940 C8GD7J 137647315 IC50 = 86.1 nM T91940 CUI30W 137647494 IC50 = 543.3 nM T91940 CV3OT8 137648131 IC50 = 803.5 nM T91940 CDSP68 137648364 IC50 = 2013.7 nM T91940 CE9KI7 137649596 IC50 > 4000 nM T91940 CW7V4A 137649894 IC50 = 350.4 nM T91940 CHLD47 137649903 IC50 = 576.8 nM T91940 C8M4KC 137650065 IC50 = 101.9 nM T91940 CK38XJ 137651046 Ki = 135 nM T91940 CX9ZD8 137651366 IC50 = 1020.9 nM T91940 CSLK59 137652206 IC50 = 95 nM T91940 C1N0FA 137652292 IC50 = 5200 nM T91940 CFZD39 137652732 IC50 = 7400 nM T91940 CU7IQ6 137653037 IC50 = 9078.2 nM T91940 CR36ZA 137653185 IC50 = 30.3 nM T91940 CR3N8X 137653273 IC50 > 40000 nM T91940 C8L4QI 137654079 IC50 = 1798.8 nM T91940 COQ34W 137654121 IC50 = 644.1 nM T91940 CEU75P 137654196 IC50 = 176.6 nM T91940 CGSX07 137654767 IC50 = 739.6 nM T91940 C1IQR5 137654865 IC50 = 4300 nM T91940 CL8W1A 137655192 IC50 = 90000 nM T91940 C1ZY5K 137655408 IC50 = 295.1 nM T91940 C1M6GP 137655507 IC50 = 3388.4 nM T91940 CPER95 137655658 IC50 = 533.3 nM T91940 CQBT10 137656275 IC50 = 591.6 nM T91940 C0PGM5 137656289 Ki = 3.5 nM T91940 CA9CU0 137657316 IC50 = 3097.4 nM T91940 C3O0BX 137657532 IC50 = 631 nM T91940 CLO1P4 137658149 IC50 = 352.4 nM T91940 CE34VH 137658343 IC50 = 792.5 nM T91940 C3N4SQ 137658444 IC50 = 857 nM T91940 C72EBT 137658527 IC50 = 2196.2 nM T91940 C5TY2U 137658918 IC50 = 1258.9 nM T91940 CK7A3W 137659231 IC50 = 1075.4 nM T91940 C1D9AJ 137659323 IC50 = 1148.2 nM T91940 C90LUW 137659427 IC50 = 119.9 nM T91940 C0Z9VM 137659462 IC50 = 3732.5 nM T91940 CH1JW4 137659577 Ki = 23 nM T91940 CCFW90 137659626 IC50 = 89.9 nM T91940 C30QFV 137660965 Ki = 3.5 nM T91940 CZY3M1 137661177 IC50 = 124000 nM T91940 C15BNL 137661289 IC50 = 2710.2 nM T91940 C7FIH9 137661665 IC50 = 431.5 nM T91940 C8CY9Q 137661720 IC50 = 154000 nM T91940 CW7HG8 145960911 IC50 > 500000 nM T91940 CC0VT3 145962411 IC50 > 50000 nM T91940 C5QIN6 145963700 IC50 > 500000 nM T91940 CPQ48B 155513088 IC50 > 200000 nM T91940 CZE29G 155514745 IC50 > 150000 nM T91940 D09SUO 5269 IC50 > 100000 nM T91940 D0E3NT 2130404 IC50 > 100000 nM T63682 D0E3TC 44259 IC50 = 2.11 nM T63682 C3VRO9 44557921 IC50 > 10000 nM T63682 C8W6IG 57395117 IC50 > 30000 nM T63682 CV63UL 67240318 IC50 > 10000 nM T63682 C1NPL0 71552941 IC50 > 30000 nM T63682 CA4PS8 71552942 IC50 > 30000 nM T63682 C2MD1Q 155513187 IC50 > 10000 nM T63682 D03DZO 11715767 IC50 > 10000 nM T63682 D0T8NU 16757525 IC50 = 126 nM T78710 D0L9QM 59568713 IC50 = 6 nM T78710 C0F4YK 2980278 IC50 = 6500 nM T78710 CNV4F5 4536383 IC50 = 290 nM T78710 C0I8GC 14985965 IC50 = 5200 nM T78710 CM75QU 49801042 IC50 = 60 nM T78710 C8LFB9 49801043 IC50 = 110 nM T78710 C8IYR7 49801044 IC50 = 220 nM T78710 C6QJX1 49802220 IC50 = 61 nM T78710 CEP69H 49802221 IC50 = 130 nM T78710 CP91TS 49802222 IC50 = 340 nM T78710 CIFZ02 49803320 IC50 = 15 nM T78710 CEP3B7 49803607 IC50 = 9 nM T78710 C1BLY0 49804185 IC50 = 96 nM T78710 C97LZE 49804478 IC50 = 34 nM T78710 C2IGB7 49804777 IC50 = 70 nM T78710 C3XQE2 52337837 IC50 = 24 nM T78710 CS4HK7 53354783 IC50 = 49 nM T78710 CJ6DK1 56970422 IC50 = 89 nM T78710 CDH38V 56970630 IC50 = 76 nM T78710 C67JVW 56970631 IC50 = 53 nM T78710 C4DMU9 56970632 IC50 = 26 nM T78710 C3RBO8 56970861 IC50 = 300 nM T78710 CJ5O6Y 56970863 IC50 = 430 nM T78710 C1DN0L 56970864 IC50 = 280 nM T78710 CRF6L7 56971088 IC50 = 790 nM T78710 CQ5IH3 56971089 IC50 = 35 nM T78710 CHN80L 57331188 IC50 = 430 nM T78710 C4E1NK 57331209 IC50 = 64 nM T78710 C8PWJ3 57331210 IC50 = 460 nM T78710 C1E3WV 57331240 IC50 = 110 nM T78710 C4WI9O 57331241 IC50 = 160 nM T78710 C68CPW 57331268 IC50 = 470 nM T78710 CD0WM9 57331302 IC50 = 61 nM T78710 CY0W1H 57331373 IC50 = 540 nM T78710 CGUA26 57331668 IC50 = 20 nM T78710 CG2V1M 59568650 IC50 = 49 nM T78710 C7FAN1 59568652 IC50 = 67 nM T78710 CM1G2P 59568656 IC50 = 32 nM T78710 CS19JW 59568702 IC50 = 12 nM T78710 CL42CH 60509567 IC50 = 140 nM T78710 CL9JR7 67516635 IC50 = 190 nM T78710 CIB4Y6 67516958 IC50 = 550 nM T78710 COH79P 67517411 IC50 = 89 nM T78710 C0WAQ6 67517817 IC50 = 330 nM T78710 C02TCR 67518221 IC50 = 920 nM T78710 CG24FU 68071359 IC50 = 75 nM T78710 CG2QU1 68071450 IC50 = 79 nM T78710 CNS57A 68071672 IC50 = 170 nM T78710 CJ8Y2W 68071788 IC50 = 170 nM T78710 CR5BI7 68071790 IC50 = 620 nM T78710 C3DZ1N 68071887 IC50 = 550 nM T78710 CKJ13C 68095253 IC50 = 440 nM T78710 C4C5PG 68431603 IC50 = 410 nM T78710 C1VIW9 68431605 IC50 >= 1000 nM T78710 CA9MK4 68432911 IC50 = 18 nM T78710 C7SC0U 68432912 IC50 >= 1000 nM T78710 CJM2Y1 69087440 IC50 = 1100 nM T78710 CZ0IC8 69087441 IC50 = 160 nM T78710 C08ZXY 69087444 IC50 = 830 nM T78710 C04OLI 69087452 IC50 = 66 nM T78710 C59HRV 69087454 IC50 = 29 nM T78710 CXV98R 69087490 IC50 = 38 nM T78710 C1XE4Q 69087494 IC50 = 450 nM T78710 CGQ40U 69087495 IC50 = 72 nM T78710 CCO97X 69087505 IC50 = 300 nM T78710 CI3A6W 69087537 IC50 = 510 nM T78710 CMA21H 69087541 IC50 = 95 nM T78710 CQF9T5 69087543 IC50 = 69 nM T78710 CVG42E 69087545 IC50 = 26 nM T78710 CX3P0T 69087562 IC50 = 250 nM T78710 CF0YK9 71449242 IC50 > 10000 nM T78710 CCX2W5 71449253 IC50 = 1900 nM T78710 C0B7ZW 71451051 IC50 = 89 nM T78710 C0L8PR 71451052 IC50 = 340 nM T78710 CE98WI 71451053 IC50 = 4200 nM T78710 C42GQM 71452880 IC50 = 4300 nM T78710 C3JZH1 71452881 IC50 = 2200 nM T78710 CKMZ80 71452882 IC50 = 12000 nM T78710 C8Q0JV 71454645 IC50 = 4600 nM T78710 CGJE74 71454646 IC50 = 3800 nM T78710 CT7EN2 71456366 IC50 = 3800 nM T78710 CE40RO 71456367 IC50 > 10000 nM T78710 C3YOV7 71456368 IC50 = 99 nM T78710 C9DN6M 71458213 IC50 > 10000 nM T78710 CYW78K 71458214 IC50 > 10000 nM T78710 CI7B2J 71458215 IC50 = 240 nM T78710 CYD4J7 71460068 IC50 > 10000 nM T78710 C89YUI 71460069 IC50 = 9400 nM T78710 CV6QH8 71461787 IC50 = 2900 nM T78710 CC92TB 71461788 IC50 = 3100 nM T78710 C1PC8B 71516677 IC50 = 120 nM T78710 C3YA4C 71603551 IC50 = 27 nM T78710 C6MZO8 71603797 IC50 = 72 nM T78710 CNGS29 71603853 IC50 = 104 nM T78710 CKY82R 71603916 IC50 = 39 nM T78710 C9J0EH 71603917 IC50 = 73 nM T78710 CT8ZS9 71603918 IC50 = 70 nM T78710 C2X3AO 71603919 IC50 = 41 nM T78710 CFTR25 71603920 IC50 = 36 nM T78710 C7BD6V 71603987 IC50 = 57 nM T78710 C98YDN 71603990 IC50 = 60 nM T78710 CQ37SD 71604125 IC50 = 86 nM T78710 C2PBS7 72375648 IC50 = 1800 nM T78710 C23VDP 72375650 IC50 = 7100 nM T78710 CTED19 72375651 IC50 > 32000 nM T78710 CRZ48N 72375747 IC50 = 1300 nM T78710 C6W8VM 72375748 IC50 = 1200 nM T78710 CU9DR1 72375749 IC50 = 610 nM T78710 CA0Y6E 72375832 IC50 = 2500 nM T78710 CT98UV 72375833 IC50 = 100000 nM T78710 CKS9M4 72375834 IC50 = 71 nM T78710 CV19HQ 72375835 IC50 = 520 nM T78710 CJ9T5X 72375921 IC50 = 1400 nM T78710 CCP0Q4 72376019 IC50 = 460 nM T78710 C3EV2U 73352607 IC50 = 1500 nM T78710 C6AN3L 73357170 IC50 = 2100 nM T78710 CM73EU 76901852 IC50 = 60 nM T78710 CLC6F8 77938792 IC50 = 49 nM T78710 CR76VN 86694482 IC50 = 300 nM T78710 CP4T5E 89619103 IC50 = 18 nM T78710 C89MLI 89619107 IC50 = 33 nM T78710 CZ1A3U 89619266 IC50 = 107 nM T78710 C7T9GQ 89633340 IC50 = 57 nM T78710 C4D3MX 89633347 IC50 = 165 nM T78710 CXPV63 89633380 IC50 = 83 nM T78710 CRWG69 89633382 IC50 = 45 nM T78710 CX4MP3 89633392 IC50 = 260 nM T78710 C5FZ4E 89633466 IC50 = 86 nM T78710 C8MN9K 89763714 IC50 = 150 nM T78710 CL4WR9 90465846 IC50 = 29 nM T78710 C3PLV0 91810383 IC50 = 27.46 nM T78710 C4O3VF 117689963 IC50 = 88 nM T78710 C0HD1T 117690173 IC50 = 50 nM T78710 CT7GW0 117690258 IC50 = 65 nM T78710 CX0DY2 117690263 IC50 = 112 nM T78710 CQF32S 117690304 IC50 = 100 nM T78710 C15QUL 117690396 IC50 = 105 nM T78710 CZGO85 117852204 IC50 = 20 nM T78710 CBD0X6 117852205 IC50 = 50 nM T78710 CN5H7Y 117852210 IC50 = 76 nM T78710 CB9X7D 117852213 IC50 = 127 nM T78710 CTKJ90 117852221 IC50 = 89 nM T78710 C3PST8 117852226 IC50 = 47 nM T78710 C75VGS 117852234 IC50 = 10.1 nM T78710 CN8G6X 117852236 IC50 = 10 nM T78710 C3SW9X 117852238 IC50 = 37 nM T78710 CO3X7N 117852239 IC50 = 308 nM T78710 C17KYZ 117852241 IC50 = 43 nM T78710 CI06AN 117852248 IC50 = 104 nM T78710 C3K8XU 117852302 IC50 = 10 nM T78710 C78VZX 117852306 IC50 = 14 nM T78710 CH31XV 117852322 IC50 = 17 nM T78710 CMS0A3 117852327 IC50 = 34 nM T78710 C04UHW 117852380 IC50 = 10 nM T78710 CQ4FJ5 117852383 IC50 = 37 nM T78710 C4U3KW 117852415 IC50 = 12 nM T78710 C52IZU 118174492 IC50 = 477.1 nM T78710 CVP6Q3 118174494 IC50 = 81.43 nM T78710 CR5J4P 118189027 IC50 = 74.74 nM T78710 CFE27D 118189030 IC50 = 66 nM T78710 CSTV63 118189049 IC50 = 463 nM T78710 C6E2VF 121305983 IC50 = 37 nM T78710 CL8P4D 121305987 IC50 = 12 nM T78710 CR0HG1 121313818 IC50 = 420 nM T78710 CO97HF 121313830 IC50 = 27 nM T78710 CCUN52 121313839 IC50 = 550 nM T78710 C4USB9 121313840 IC50 = 4 nM T78710 C1GPN7 121313866 IC50 = 350 nM T78710 CML4Z3 121313870 IC50 = 250 nM T78710 CWC64Z 121313891 IC50 = 95 nM T78710 C37BWZ 121313899 IC50 = 620 nM T78710 CC9A1P 121313903 IC50 = 510 nM T78710 CA5L4N 121313914 IC50 = 54 nM T78710 C0VQ4K 121313943 IC50 = 340 nM T78710 CD6Z2S 121313948 IC50 = 11 nM T78710 C5TJ0N 121313953 IC50 = 130 nM T78710 C1H8OV 121313959 IC50 = 430 nM T78710 CTD80X 121313965 IC50 = 490 nM T78710 CU4CW1 121313969 IC50 = 17 nM T78710 CFP26R 121313971 IC50 = 260 nM T78710 CNT7G1 121313972 IC50 = 270 nM T78710 CC1G3N 121313978 IC50 = 77 nM T78710 C8ZC5L 121313982 IC50 = 430 nM T78710 CR74PF 121313995 IC50 = 190 nM T78710 CTD40H 121314002 IC50 = 68 nM T78710 CQFC86 121314009 IC50 = 56 nM T78710 C8I2PZ 121314020 IC50 = 59 nM T78710 C7QK2C 121314021 IC50 = 180 nM T78710 CJT43I 121314036 IC50 = 42 nM T78710 C8PT6Y 121314045 IC50 = 20 nM T78710 CH8S4J 121314048 IC50 = 51 nM T78710 CFW68T 121314052 IC50 = 130 nM T78710 CP13EB 121314068 IC50 = 120 nM T78710 C1BO8D 121483467 IC50 = 13 nM T78710 C52XCY 122188482 IC50 = 120 nM T78710 C2XJ7S 122188483 IC50 = 43 nM T78710 CUF9Y6 122188484 IC50 > 3000 nM T78710 CPW3L7 122188565 IC50 = 46 nM T78710 CSDG34 122188566 IC50 = 130 nM T78710 C1F2GQ 122188567 IC50 = 29 nM T78710 C49ACM 122188568 IC50 = 850 nM T78710 CCQ2U5 122188569 IC50 = 16 nM T78710 CZ07LD 122191612 IC50 = 15 nM T78710 C53LVE 122191613 IC50 = 14 nM T78710 CX5J6C 122191614 IC50 = 14 nM T78710 CWS5J3 122191615 IC50 = 9 nM T78710 CO97EW 127043792 IC50 = 9 nM T78710 CTW30M 127043793 IC50 = 35 nM T78710 C3XME6 127043966 IC50 = 43 nM T78710 CK5AB9 127043967 IC50 = 11 nM T78710 C90TWS 127043968 IC50 = 20 nM T78710 CBH5T4 127043969 IC50 = 14 nM T78710 C2OGR1 127044121 IC50 = 32 nM T78710 C2EVN7 127044122 IC50 = 7 nM T78710 CTX6M9 127044123 IC50 = 19 nM T78710 CLNO38 127044124 IC50 = 17 nM T78710 CY53KO 127044257 IC50 = 31 nM T78710 CY14VE 130449668 IC50 = 47 nM T78710 C7HB2T 130449692 IC50 = 17 nM T78710 CZB60C 130449716 IC50 = 65 nM T78710 C70SUN 130449733 IC50 = 420 nM T78710 CZCT84 130449749 IC50 = 88 nM T78710 C9YSZ8 130449791 IC50 = 5 nM T78710 CIV73D 132020378 IC50 = 28 nM T78710 CP9L2O 132020426 IC50 = 38 nM T78710 CR6I1X 134134165 IC50 = 140 nM T78710 CIGL40 134145890 IC50 = 205 nM T78710 CA25UM 137351045 IC50 = 6.6 nM T78710 CBR0X1 137632751 IC50 = 901 nM T78710 CVH35W 137633042 IC50 = 6400 nM T78710 CH43XI 137633091 IC50 = 7600 nM T78710 CE6ZM1 137635237 IC50 = 5100 nM T78710 CJX8N5 137640241 IC50 = 41 nM T78710 C4MN6W 137643261 IC50 = 1000 nM T78710 COH10Y 137651081 IC50 = 10 nM T78710 C1ZH9J 137659238 IC50 = 570 nM T78710 CYI45R 137660122 IC50 = 1050 nM T78710 C7H2LV 137660844 IC50 > 2000 nM T78710 C29DMS 137661489 IC50 > 2000 nM T78710 C7Q6MF 145951374 IC50 = 35 nM T78710 CX2UH4 145952348 IC50 = 62 nM T78710 CVS48W 145952572 IC50 = 86 nM T78710 CBO52Q 145954980 IC50 = 100 nM T78710 CJ5GW3 145956273 IC50 = 17000 nM T78710 C0LJB1 145956360 IC50 = 1300 nM T78710 CB8S9C 145957865 IC50 = 61 nM T78710 CQ19NA 145958506 IC50 = 398.11 nM T78710 CZK51T 145958678 IC50 = 104 nM T78710 C5N2KJ 155529339 IC50 = 8.8 nM T78710 C1DV5G 155552667 IC50 = 65 nM T78710 CSI0H9 155553919 IC50 = 6.2 nM T78710 CNOP56 155557940 Ki = 2 nM T78710 CD38PJ 155559250 IC50 = 6.6 nM T78710 D05LBC 44123657 IC50 = 240 nM T28052 D0L5WM 2157 IC50 = 99000 nM T28052 D0X5SD 3117 IC50 = 10000 nM T28052 D00SUC 74766595 IC50 = 13 nM T28052 D01WHH 90216982 IC50 < 100 nM T28052 D03POM 132054530 IC50 = 65 nM T28052 D05CCY 77106319 IC50 = 100 nM T28052 D0G8QR 76282772 IC50 < 100 nM T28052 D0GH8J 90204862 IC50 < 100 nM T28052 D0K4LW 90205053 IC50 < 100 nM T28052 D0NM3B 121279569 IC50 = 7200 nM T28052 D0PQ5P 117637389 IC50 = 6700 nM T28052 D0T8YT 121279737 IC50 = 60 nM T28052 CB9CG6 1742 IC50 = 13000 nM T28052 C25LHT 125134 IC50 = 26000 nM T28052 CO71PD 610500 IC50 = 7000 nM T28052 C2OS6J 651205 IC50 = 237 nM T28052 CMKP07 736587 IC50 = 878 nM T28052 CU1M9F 848720 IC50 = 25000 nM T28052 C3RTG1 992337 IC50 = 83000 nM T28052 CE4HM8 1032885 IC50 = 3800 nM T28052 C8G2LC 1736340 IC50 = 5000 nM T28052 C5BZF0 2819027 IC50 = 649 nM T28052 C6RA7F 3126079 IC50 = 13000 nM T28052 C83LHI 3239476 IC50 = 20 nM T28052 CWG81U 5429178 IC50 = 4200 nM T28052 CLQ21I 5852401 IC50 = 64000 nM T28052 C6LCX3 6260040 IC50 = 15000 nM T28052 CTC90M 6519698 IC50 = 251.19 nM T28052 CUA1X4 7099919 IC50 = 25000 nM T28052 C2DBN5 46899607 IC50 = 13000 nM T28052 C3NE8O 46931242 IC50 > 10000 nM T28052 CM07QJ 53380011 IC50 = 18000 nM T28052 C2HXA1 53380104 IC50 = 4000 nM T28052 CCF24D 54149635 IC50 = 48000 nM T28052 CZ0O6U 54684458 IC50 > 25000 nM T28052 CK8GB4 54694513 IC50 > 25000 nM T28052 CLQ01M 54720991 IC50 = 6700 nM T28052 CTV18U 54731416 IC50 > 25000 nM T28052 CU8AX0 55281807 IC50 = 10400 nM T28052 C2P7SD 56577044 IC50 > 10000 nM T28052 CD57TH 56666474 IC50 = 571000 nM T28052 CMO90J 56997255 IC50 = 46000 nM T28052 CXY3E4 57720618 IC50 > 30000 nM T28052 C0WX5O 70679311 IC50 > 10000 nM T28052 CLZ7P4 70702119 IC50 = 26000 nM T28052 CW1GP2 70702121 IC50 = 41000 nM T28052 CY21XA 70702122 IC50 = 30000 nM T28052 CEW3R6 71598546 IC50 > 30000 nM T28052 C14GIV 71735687 IC50 = 100000 nM T28052 CM02VN 71735839 IC50 = 64000 nM T28052 C4WS1H 71735840 IC50 = 93000 nM T28052 CT4YO5 71735841 IC50 = 35000 nM T28052 C2ZFM8 71735842 IC50 = 55000 nM T28052 CI5W0K 71735843 IC50 = 55000 nM T28052 CUD65X 73333125 IC50 > 10000 nM T28052 CHQ18I 73333126 IC50 > 10000 nM T28052 C9UDN1 73333127 IC50 > 10000 nM T28052 C9K1NV 73333128 IC50 > 10000 nM T28052 C4UE6G 73333129 IC50 > 10000 nM T28052 CV2SJ4 73333225 IC50 > 10000 nM T28052 CF8HO3 73333226 IC50 > 10000 nM T28052 CVH9F0 73333227 IC50 > 10000 nM T28052 C4PYG2 73333229 IC50 > 10000 nM T28052 CBJC52 73333322 IC50 > 10000 nM T28052 CFY18G 73333510 IC50 = 210000 nM T28052 CVEN67 73334066 IC50 > 10000 nM T28052 CYL3M7 73334067 IC50 > 10000 nM T28052 C6T7YX 73334068 IC50 > 10000 nM T28052 C70XCT 73334069 IC50 > 10000 nM T28052 C8QWP1 73334070 IC50 > 10000 nM T28052 CR98DL 73334157 IC50 > 10000 nM T28052 CJD9C1 73334158 IC50 > 10000 nM T28052 CLRM71 73334159 IC50 > 10000 nM T28052 C43NER 73334160 IC50 > 10000 nM T28052 CD2HX4 73334161 IC50 > 10000 nM T28052 CC89FN 73334162 IC50 > 10000 nM T28052 COV3R1 73334262 IC50 > 10000 nM T28052 CZD0N1 73334263 IC50 > 10000 nM T28052 CU3KG0 73334264 IC50 > 10000 nM T28052 CMLV27 73334265 IC50 > 10000 nM T28052 CD0VK7 73334266 IC50 > 10000 nM T28052 C1SGJ3 73334267 IC50 > 10000 nM T28052 C3PYF5 73334361 IC50 > 10000 nM T28052 C8H9JF 73334363 IC50 > 10000 nM T28052 C8XE1J 73334364 IC50 > 10000 nM T28052 CN40ZI 73334365 IC50 > 10000 nM T28052 CF9GA5 73334366 IC50 > 10000 nM T28052 C69WLM 73334479 IC50 > 10000 nM T28052 CG32QB 73334480 IC50 > 10000 nM T28052 CVE0S2 73334481 IC50 > 10000 nM T28052 C2S8XN 73334482 IC50 > 10000 nM T28052 CXJP87 73334483 IC50 > 10000 nM T28052 C57KSE 73334484 IC50 > 10000 nM T28052 CAQ18T 73334592 IC50 > 10000 nM T28052 CA67YG 73334593 IC50 > 10000 nM T28052 CNS84D 73334594 IC50 > 10000 nM T28052 C93HWE 73334595 IC50 > 10000 nM T28052 C87UBE 73334596 IC50 > 10000 nM T28052 CKSY83 73334696 IC50 > 10000 nM T28052 C36QHM 73334697 IC50 > 10000 nM T28052 CF63HU 73334698 IC50 > 10000 nM T28052 CQBX27 73334699 IC50 > 10000 nM T28052 C0OW1V 73334700 IC50 > 10000 nM T28052 CG80NF 73349257 IC50 > 10000 nM T28052 COY1J2 73349259 IC50 > 10000 nM T28052 CNO9Z5 73350843 IC50 > 10000 nM T28052 CN5B4O 73352277 IC50 = 110000 nM T28052 C8U0ZX 73352326 IC50 > 10000 nM T28052 C2OXQ5 76314887 IC50 > 30000 nM T28052 C3X7EW 76314888 IC50 > 30000 nM T28052 C1YKN5 76314889 IC50 > 30000 nM T28052 C4E1BN 76318504 IC50 > 30000 nM T28052 CF76CT 76318505 IC50 > 30000 nM T28052 CLVA91 76318506 IC50 > 30000 nM T28052 C9LNK4 76318507 IC50 > 30000 nM T28052 CL87KC 76318508 IC50 > 30000 nM T28052 CET23F 76318509 IC50 > 30000 nM T28052 C01JLF 76322168 IC50 > 30000 nM T28052 C2SEM0 76322169 IC50 > 30000 nM T28052 CRH48X 76322170 IC50 > 30000 nM T28052 C5CZV2 76325789 IC50 > 30000 nM T28052 CS6GL0 76333019 IC50 > 30000 nM T28052 C7IUX5 76333020 IC50 > 30000 nM T28052 CZC8W2 76336632 IC50 > 30000 nM T28052 CYQ0B9 76336633 IC50 > 30000 nM T28052 CK2N0L 76336634 IC50 > 30000 nM T28052 CS4W5I 76336635 IC50 > 30000 nM T28052 CM6H9O 76336636 IC50 > 30000 nM T28052 C3GZ6W 78425985 IC50 = 55 nM T28052 C8X6DL 78425992 IC50 = 214 nM T28052 C6IJN1 78426128 IC50 = 324 nM T28052 C3ABF9 78426132 IC50 = 3090 nM T28052 C0R5DO 78426278 IC50 = 2240 nM T28052 CX49NK 78426282 IC50 = 15 nM T28052 CPR02W 78426283 IC50 = 712 nM T28052 CMR52S 78426698 IC50 = 10 nM T28052 C6ZNK4 78426702 IC50 = 9.2 nM T28052 C1G6MS 78426838 IC50 = 63.2 nM T28052 C8L5JM 78426839 IC50 = 18 nM T28052 C3E2QY 78426985 IC50 = 10 nM T28052 CJU0V3 78427123 IC50 = 18.2 nM T28052 CGM14B 82273434 IC50 = 9.3 nM T28052 CIG3E9 83672127 IC50 = 220 nM T28052 CS4Q1F 86268882 IC50 < 100 nM T28052 C8WA4M 86725535 IC50 = 550 nM T28052 C8MGN0 86725568 IC50 = 4 nM T28052 C9IYE0 90204662 IC50 = 12 nM T28052 CB3I6M 90204812 IC50 = 240 nM T28052 CHV05N 90204861 IC50 = 1700 nM T28052 C6PI4M 90204893 IC50 = 77 nM T28052 CU8SJ5 90204921 IC50 = 6 nM T28052 C5A3VQ 90204958 IC50 = 250 nM T28052 CIY20E 90204966 IC50 = 75 nM T28052 C6DA2O 90204997 IC50 = 270 nM T28052 CO8UQ0 90205153 IC50 = 18 nM T28052 C5ST7H 90205231 IC50 = 32 nM T28052 CJ37CO 90205235 IC50 = 100 nM T28052 CQV07L 90205291 IC50 = 44 nM T28052 CJ5E4U 90205326 IC50 = 19 nM T28052 C5W7FL 90205353 IC50 = 3 nM T28052 C7ZVG4 90205376 IC50 = 430 nM T28052 CM2NA1 90205425 IC50 = 38 nM T28052 CB7Z0A 90205426 IC50 = 32 nM T28052 C2T4RD 90205719 IC50 = 29 nM T28052 C9H8PV 90211058 IC50 = 180 nM T28052 C1GBT5 90225370 IC50 = 100 nM T28052 CFX8E0 90407594 IC50 = 100 nM T28052 CJ9OZ4 90407809 IC50 = 100 nM T28052 C5LDR2 90407841 IC50 < 100 nM T28052 CSZ96D 90418518 IC50 > 25000 nM T28052 CGY5R3 90419531 IC50 = 27.5 nM T28052 C37KLX 90419541 IC50 = 5.3 nM T28052 CSOE73 90419617 IC50 = 29.3 nM T28052 CD9FZ8 90419692 IC50 = 13.1 nM T28052 CWGA54 90420023 IC50 = 21.1 nM T28052 CDU6J5 90442347 IC50 = 1180 nM T28052 C1UVE9 90442348 IC50 = 206 nM T28052 CV1RA9 90454565 IC50 = 5.6 nM T28052 CQE35S 90454567 IC50 = 12.3 nM T28052 C8H0ZM 90454574 IC50 = 13.3 nM T28052 CM2Y9N 90454575 IC50 = 13.9 nM T28052 CS12UL 90454577 IC50 = 11.1 nM T28052 CH39EW 90454586 IC50 = 28.3 nM T28052 C2EM8R 90454601 IC50 = 31.6 nM T28052 C2V3NY 90454615 IC50 = 319 nM T28052 CR3NW4 90454619 IC50 = 10.4 nM T28052 CZ0S4H 90454621 IC50 = 17.5 nM T28052 CSGN26 90454622 IC50 = 20.1 nM T28052 CS8B9I 90454628 IC50 = 28.9 nM T28052 C1V6WM 90454630 IC50 = 20.3 nM T28052 C8L0ZW 90454642 IC50 = 35.9 nM T28052 C90MQW 90454664 IC50 = 13.8 nM T28052 CF3A8C 90454673 IC50 = 18 nM T28052 CDX3P0 90454683 IC50 = 12.8 nM T28052 CQL45I 90454688 IC50 = 15.9 nM T28052 CB9G2Q 90454701 IC50 = 29 nM T28052 CKNT83 90454710 IC50 = 10.1 nM T28052 CAZY58 90454746 IC50 = 24 nM T28052 C7MXT5 90454779 IC50 = 15 nM T28052 CQ7Z5O 90454792 IC50 = 6.2 nM T28052 C9KR0V 90454795 IC50 = 5400 nM T28052 CWJ91C 90454806 IC50 = 24.7 nM T28052 C7A9GN 90454817 IC50 = 20.4 nM T28052 CN1MC4 91663282 IC50 = 2.3 nM T28052 C2S1AO 110264830 IC50 = 260 nM T28052 CA1OC5 118908372 IC50 = 11.2 nM T28052 C7TBE9 118908379 IC50 = 14 nM T28052 C13SUQ 118908442 IC50 = 15.5 nM T28052 CJVK69 119081409 IC50 < 500 nM T28052 C1RLA6 121279427 IC50 = 458 nM T28052 C39CFL 121279428 IC50 = 357 nM T28052 CC3JR1 121279532 IC50 = 251 nM T28052 CR20FE 121279544 IC50 = 1100 nM T28052 CA2K1G 121279570 IC50 = 128 nM T28052 C18TCO 121279610 IC50 > 25000 nM T28052 CQSZ74 121279659 IC50 = 8900 nM T28052 CUK15I 121279677 IC50 = 469 nM T28052 C4AIZ2 121279678 IC50 = 265 nM T28052 C2GIN5 121279684 IC50 = 878 nM T28052 CYM4R2 121279687 IC50 = 897 nM T28052 C50ZPC 121279690 IC50 = 1500 nM T28052 C9NZQ3 121279698 IC50 = 2600 nM T28052 CL9DM4 121279700 IC50 = 122 nM T28052 CR9XM8 121279703 IC50 = 105 nM T28052 C0QON3 121279710 IC50 = 727 nM T28052 CON4V9 121279730 IC50 = 14300 nM T28052 C9O7PB 121488114 IC50 = 50 nM T28052 C5IZD1 122181577 IC50 = 4300 nM T28052 CY3CG7 122181578 IC50 = 53000 nM T28052 CSR0K5 122181579 IC50 = 6300 nM T28052 CQ57MD 122181580 IC50 = 1800 nM T28052 CQ83MR 122181581 IC50 = 7800 nM T28052 C4GU9P 122181582 IC50 = 8900 nM T28052 CRM93S 122181583 IC50 = 79 nM T28052 CU57QX 122181584 IC50 = 3300 nM T28052 CIM8C2 122181585 IC50 = 14000 nM T28052 CQA0H7 122181586 IC50 = 19000 nM T28052 C9QVZ5 122181587 IC50 = 4500 nM T28052 CJQ91K 122181588 IC50 = 3100 nM T28052 CICZ91 122181589 IC50 = 63000 nM T28052 C56BUC 122181590 IC50 = 21000 nM T28052 C63NWD 127030711 IC50 > 10000 nM T28052 CN16WB 127030937 IC50 = 100 nM T28052 CFZ3S6 127031895 IC50 = 41000 nM T28052 CDC17F 127032730 IC50 = 1000 nM T28052 CL38FP 127033048 IC50 = 100 nM T28052 CWP07A 129606887 IC50 = 1800 nM T28052 C7AVR9 131637453 IC50 = 1577000 nM T28052 C3AL6C 132070185 IC50 = 14600 nM T28052 C3VG6R 132070189 IC50 > 25000 nM T28052 CDJ50A 132070206 IC50 = 198 nM T28052 C6ST2Z 132472258 IC50 = 590 nM T28052 CDZ4H0 132472263 IC50 = 670 nM T28052 C5OSR0 133053810 IC50 = 1400 nM T28052 CEV3A1 133053816 IC50 = 71000 nM T28052 CYD7R0 133053821 IC50 = 290 nM T28052 CAZ6V1 133053881 IC50 = 22000 nM T28052 CGAK71 133053891 IC50 = 690 nM T28052 CM6KI8 135487489 IC50 = 2300 nM T28052 CT4O5U 135567037 IC50 = 180000 nM T28052 CC4H1N 135567038 IC50 = 23000 nM T28052 CQBH95 135567040 IC50 = 240000 nM T28052 CP6IH9 135567041 IC50 = 45000 nM T28052 C8HMG2 135567042 IC50 = 52000 nM T28052 CT0DW5 136048747 IC50 < 100 nM T28052 CXW0S7 136048748 IC50 < 100 nM T28052 CJ91RY 136048749 IC50 < 100 nM T28052 CM2VE8 136165229 IC50 = 160 nM T28052 C1H9NK 136959977 IC50 < 100 nM T28052 CLUX03 137174251 IC50 > 10000 nM T28052 C91JZQ 137321153 IC50 = 100 nM T28052 C0D7SY 137349487 IC50 = 83000 nM T28052 CFM25A 137632245 IC50 = 430 nM T28052 C8B4IH 137632294 IC50 > 25000 nM T28052 CG6I9H 137633084 IC50 > 25000 nM T28052 C4PN0K 137634783 IC50 = 204 nM T28052 C8S5FP 137635888 IC50 > 25000 nM T28052 C8RGO2 137636770 IC50 > 25000 nM T28052 C6KMJ9 137638363 EC50 = 6500 nM T28052 CT1L5K 137639466 IC50 > 25000 nM T28052 C7E9FR 137640082 IC50 = 4500 nM T28052 CIV98W 137645322 IC50 > 25000 nM T28052 CB04DM 137646808 IC50 > 25000 nM T28052 CC9IH3 137647924 IC50 > 25000 nM T28052 CM2Z0N 137653564 IC50 > 25000 nM T28052 C3XEA6 137654812 IC50 > 25000 nM T28052 CY2Q8D 137659279 IC50 > 25000 nM T28052 CGM39L 137661457 IC50 = 3300 nM T28052 C1ANF3 138518187 IC50 = 25 nM T28052 C97JVF 145948622 IC50 = 5050 nM T28052 C9XO4M 145948655 IC50 = 6740 nM T28052 CHP2V5 145948690 IC50 > 50000 nM T28052 CLD12N 145949023 IC50 = 12900 nM T28052 C5GM0U 145949030 IC50 > 50000 nM T28052 C4QC5Y 145960532 IC50 = 198000 nM T28052 C8HPT2 145961258 IC50 = 1146000 nM T28052 C9FGU1 145961684 IC50 = 844000 nM T28052 CZ0OC7 145962144 IC50 = 12600 nM T28052 CF4ME6 145962269 IC50 = 37000 nM T28052 CZP8B7 145962316 IC50 = 218000 nM T28052 CJGC76 145962553 IC50 = 166000 nM T28052 CK3DZ7 145962837 IC50 = 2305000 nM T28052 CVU6M3 145962898 IC50 = 223000 nM T28052 C3RB8P 145963156 IC50 = 198000 nM T28052 CK96HI 145963214 IC50 = 533000 nM T28052 C81CRJ 145963620 IC50 = 314000 nM T28052 C2WKX0 145963644 IC50 = 1310000 nM T28052 C0GX1R 145985174 IC50 = 700 nM T28052 C0UEA8 145992575 IC50 = 320 nM T28052 CO5BA1 155511789 IC50 = 65.3 nM T28052 C73XKF 155513277 IC50 = 3800 nM T28052 C4F5PK 155517603 IC50 = 13 nM T28052 C7HGZ0 155518256 IC50 = 170 nM T28052 C60IFL 155522231 IC50 = 76.6 nM T28052 CCFX38 155528399 IC50 = 8940 nM T28052 CNY86X 155531371 IC50 = 230 nM T28052 CKM19A 155531373 IC50 = 5300 nM T28052 CPM37U 155533785 IC50 = 7.9 nM T28052 C1WZN6 155534870 IC50 = 70 nM T28052 C6N9HT 155542131 IC50 = 400 nM T28052 C9H8CB 155543083 IC50 > 25000 nM T28052 CSW87N 155543284 IC50 = 9.5 nM T28052 C4YBT0 155543964 IC50 = 11.9 nM T28052 CIM7D4 155548682 IC50 = 22.7 nM T28052 C35AFD 155549271 IC50 = 11 nM T28052 CFR06L 155551969 IC50 = 4.37 nM T28052 CD24ZA 155556847 IC50 = 179 nM T28052 C50IJC 155560285 IC50 > 25000 nM T28052 CLXJ58 155560773 IC50 = 22500 nM T28052 CNF14B 155565224 IC50 = 700 nM T28052 D07IOY 10365 IC50 = 760 nM T28052 D08IZY 3080614 IC50 = 250000 nM T28052 D0B2WZ 15331 IC50 = 2200000 nM T28052 D0I0XA 91810435 IC50 = 3200 nM T28052 D0S3DD 56963315 IC50 = 110000 nM T28052 D0W9RR 57339144 IC50 > 10000 nM T09544 D02NDV 439357 IC50 = 50000000 nM T09544 CGRE80 23651530 IC50 > 5000000 nM T09544 C5PRE0 25022444 IC50 = 313000 nM T09544 CSH54Y 44586823 IC50 > 5000000 nM T09544 C4ZAV3 44586861 IC50 > 5000000 nM T09544 CH6L3X 44586862 IC50 = 5000000 nM T09544 CTM7I3 44586863 IC50 = 5000000 nM T09544 C62VSK 44586864 IC50 > 5000000 nM T09544 CS9KL5 44586891 IC50 = 5000000 nM T09544 CJO0Y3 44586892 IC50 > 5000000 nM T09544 CGB59A 44586893 IC50 > 5000000 nM T09544 C1KTE2 44586894 IC50 > 5000000 nM T09544 CTZ16G 44586895 IC50 > 5000000 nM T09544 CY60FG 44586921 IC50 = 5000000 nM T09544 CUEA45 44586922 IC50 > 5000000 nM T09544 C0PC4W 44586923 IC50 = 5000000 nM T09544 CITZ01 44586924 IC50 = 2500000 nM T09544 C9Q6RH 44586925 IC50 > 5000000 nM T09544 CSVU02 44586950 IC50 > 5000000 nM T09544 CC5XY3 44586951 IC50 = 5000000 nM T09544 CL8WK0 44586952 IC50 = 2500000 nM T09544 CZ17UD 44586953 IC50 > 5000000 nM T09544 C1FYD6 44586954 IC50 > 5000000 nM T09544 CSM0P1 44586984 IC50 > 5000000 nM T09544 C5N4IP 44586985 IC50 = 600000 nM T09544 CBN67X 44586986 IC50 = 300000 nM T09544 CI4T9W 44586987 IC50 = 600000 nM T09544 C92USB 44586988 IC50 > 5000000 nM T09544 C1GJF9 44586989 IC50 = 300000 nM T09544 C5WJG0 44586990 IC50 = 2500000 nM T09544 CCU5M9 44587042 IC50 = 5000000 nM T09544 CL5M9D 44587043 IC50 = 300000 nM T09544 CQ4VC3 44587044 IC50 = 300000 nM T09544 CJGP86 44587045 IC50 > 5000000 nM T09544 D0K8XC 6134 IC50 = 800000 nM T85223 CXI63Y 3468 IC50 = 350 nM T85223 CER2N8 303856 IC50 > 100000 nM T85223 C1VT7G 315023 IC50 > 100000 nM T85223 CW94ZG 332819 IC50 > 100000 nM T85223 CC94ZO 2829313 IC50 > 300000 nM T85223 C9YFD0 10016842 IC50 > 100000 nM T85223 C4ETJ5 11507180 IC50 > 100000 nM T85223 CH41DP 12240669 IC50 > 100000 nM T85223 C8LOW5 44392232 IC50 > 100000 nM T85223 CZF90T 44392260 IC50 > 100000 nM T85223 CGJ3R2 54727893 IC50 > 100000 nM T85223 CBP71N 72204354 IC50 > 100000 nM T85223 C90WSF 122189950 IC50 > 100000 nM T85223 C4K3FQ 122189951 IC50 > 100000 nM T85223 CN06CL 122189952 IC50 > 100000 nM T85223 CT5X7W 122189953 IC50 > 100000 nM T85223 CG7QR3 122189954 IC50 > 100000 nM T85223 CCH93W 122189956 IC50 > 100000 nM T85223 CK2Z7A 122189957 IC50 > 100000 nM T85223 C1E4QR 122189958 IC50 > 100000 nM T85223 CC5H8Z 122189961 IC50 > 100000 nM T85223 C9VH1T 122189962 IC50 > 100000 nM T85223 C0UO8I 122189965 IC50 > 100000 nM T85223 CWJ63I 122189966 IC50 > 100000 nM T85223 CSXH56 122189967 IC50 > 100000 nM T85223 CUSD28 122189968 IC50 > 100000 nM T85223 CV87MX 122189969 IC50 > 100000 nM T85223 CBT57O 122189970 IC50 > 100000 nM T85223 CV0T3C 122189971 IC50 > 100000 nM T85223 CXI6M4 122189972 IC50 > 100000 nM T85223 CIJ16M 122189973 IC50 > 100000 nM T85223 CH5NK2 122189974 IC50 > 100000 nM T85223 C4DAW3 122189975 IC50 > 100000 nM T85223 CD2X8M 122189976 IC50 > 100000 nM T85223 C5JLT2 122189978 IC50 > 100000 nM T85223 C1BOP9 122189979 IC50 > 100000 nM T85223 CR6C9A 122189980 IC50 > 100000 nM T85223 CZI6C2 122189981 IC50 > 100000 nM T85223 C8KYD4 122190086 IC50 = 30200 nM T85223 C1UV3C 122190087 IC50 = 27900 nM T85223 CR1HZ8 122190088 IC50 > 100000 nM T85223 CTLI97 122190089 IC50 = 87000 nM T85223 C79XCY 122190090 IC50 > 100000 nM T85223 CP5G7U 135406878 IC50 > 100000 nM T85223 C6CV9R 135419769 IC50 > 100000 nM T85223 CE9X0V 135433415 IC50 > 100000 nM T85223 CEK6W2 135446332 IC50 > 100000 nM T85223 CDCV97 135446971 IC50 > 100000 nM T85223 C4L0WU 135483599 IC50 > 100000 nM T85223 CRJ3H1 135520683 IC50 > 100000 nM T85223 CL1N4E 135765525 IC50 > 100000 nM T85223 CMB6O2 136094868 IC50 > 100000 nM T85223 C8KMW2 136094876 IC50 = 67600 nM T85223 CC1Z4M 136094877 IC50 > 100000 nM T85223 C23OFV 136094878 IC50 > 100000 nM T85223 CR3C8I 136094880 IC50 > 100000 nM T85223 CM5RQ7 136094882 IC50 = 62600 nM T85223 CEZ21O 136094884 IC50 > 100000 nM T85223 CLYM32 136094885 IC50 = 58900 nM T85223 D0NS0E 220188 IC50 > 100000 nM T86130 D0Q5LF 9961766 IC50 = 0.3 nM T86130 D02WII 9912743 IC50 = 0.13 nM T86130 D0K0NP 9812185 IC50 > 100000 nM T86130 CDOC86 303776 IC50 > 1000 nM T86130 C4U0BM 1878893 IC50 > 20000 nM T86130 CM89KX 6605251 IC50 = 0.037 nM T86130 C21AGH 9799402 IC50 = 17 nM T86130 C5JSA4 9801270 IC50 = 34.9 nM T86130 C70QDG 9801659 IC50 = 5000 nM T86130 CY2NE9 9803540 IC50 = 165 nM T86130 CL9IP5 9804331 IC50 = 95 nM T86130 CTZW25 9806910 IC50 = 32 nM T86130 CD60TR 9807600 IC50 = 0.2 nM T86130 CI51MD 9807891 IC50 = 24.5 nM T86130 CK6A0I 9808598 IC50 = 36 nM T86130 CCJ07G 9822539 IC50 = 19.8 nM T86130 C2TK9G 9822773 IC50 = 3.9 nM T86130 CCI0Z3 9824271 IC50 = 0.05 nM T86130 C4KMF1 9824454 IC50 = 604 nM T86130 C2YHE9 9828124 IC50 = 1 nM T86130 CL6EU1 9828131 IC50 = 300 nM T86130 C1OP9I 9828979 EC50 > 100000 nM T86130 C6QE2T 9829096 IC50 = 12 nM T86130 C7J3ZW 9847562 IC50 = 1.4 nM T86130 C13KPA 9848051 Ki = 1.995 nM T86130 C04PAT 9849697 IC50 = 15.4 nM T86130 C2XD7P 9851886 IC50 = 6 nM T86130 CN1R0K 9852055 IC50 = 7.1 nM T86130 CI8UN0 9867771 IC50 = 2.1 nM T86130 C53EJZ 9868509 IC50 = 454 nM T86130 C15BDL 9870319 IC50 = 8 nM T86130 C2ZAK6 9870468 IC50 = 5 nM T86130 CE31YU 9891780 IC50 = 1.5 nM T86130 CW30AB 9911200 IC50 = 27 nM T86130 CKG91P 9911524 IC50 = 100 nM T86130 CA03MS 9912398 IC50 = 18 nM T86130 CA0ZG4 9913409 IC50 = 0.48 nM T86130 CLS3T2 9913547 IC50 = 66 nM T86130 CR8NU2 9915431 IC50 = 68 nM T86130 C16EYF 9916018 IC50 = 85 nM T86130 C3BZQ8 9916723 IC50 = 2 nM T86130 CGY61A 9917020 IC50 = 5.4 nM T86130 C2E9MH 9919150 IC50 = 824000 nM T86130 CCPD70 9927009 IC50 > 100000 nM T86130 CTKJ10 9929652 IC50 = 11 nM T86130 CV6S2B 9933786 IC50 = 2.4 nM T86130 CJU4Z8 9935155 IC50 = 0.39 nM T86130 CGKR03 9938832 IC50 = 2 nM T86130 C8UN5M 9951053 IC50 = 460 nM T86130 CUH19P 9951966 IC50 = 60.6 nM T86130 CRXG24 9960917 IC50 = 1.3 nM T86130 CKB08G 9981351 Ki = 316.23 nM T86130 C94BYU 9982665 Ki = 3.981 nM T86130 C9B2PM 9984709 IC50 = 40 nM T86130 C8AJ2G 9985610 IC50 = 0.5 nM T86130 C91KYI 9985909 IC50 = 0.08 nM T86130 CS9I1B 9985993 IC50 = 1700 nM T86130 CQRV24 10008981 IC50 = 8.1 nM T86130 C47PTG 10028612 IC50 = 48 nM T86130 CO61SR 10052003 IC50 = 0.25 nM T86130 C8TE7O 10052250 IC50 = 0.42 nM T86130 C5PU7I 10053671 IC50 = 0.25 nM T86130 CE74SG 10074117 IC50 = 0.39 nM T86130 CALU36 10075519 IC50 = 0.34 nM T86130 CZ91QA 10076211 IC50 = 0.1 nM T86130 CB7P1K 10076717 IC50 = 0.1 nM T86130 C9E3JX 10076744 IC50 = 3.2 nM T86130 CL53YI 10077841 IC50 = 5 nM T86130 C71AIN 10077862 IC50 = 11 nM T86130 C6ZN8C 10097891 Ki = 0.5012 nM T86130 CYQE69 10098004 IC50 = 0.27 nM T86130 C2UY1Z 10099823 IC50 = 0.13 nM T86130 CG9MW5 10100699 IC50 = 0.74 nM T86130 C95XMW 10113895 IC50 = 16 nM T86130 C3YZ2N 10116180 IC50 = 287 nM T86130 C2UW7M 10116963 IC50 = 419 nM T86130 CL3JQ0 10117970 IC50 = 1.2 nM T86130 CHWL67 10118022 IC50 = 10 nM T86130 CL2Z0P 10118913 IC50 = 0.48 nM T86130 C8WS2G 10119516 IC50 = 6.6 nM T86130 CG9U5C 10120896 IC50 = 1.94 nM T86130 CFP37Q 10128116 IC50 = 1.1 nM T86130 CK1C9H 10128662 IC50 = 39 nM T86130 C90JVX 10128813 IC50 = 1.64 nM T86130 CQ1YJ7 10138062 IC50 = 226 nM T86130 CVPQ90 10139365 IC50 = 90 nM T86130 C2FJ7D 10141277 IC50 = 5.7 nM T86130 CLG5S1 10141712 IC50 = 382 nM T86130 CEY8L9 10142180 IC50 = 10000 nM T86130 COL89Y 10142181 IC50 = 4700 nM T86130 CH54AE 10142853 IC50 = 7200 nM T86130 CDKH03 10142854 IC50 = 550 nM T86130 CF3IG8 10143847 IC50 = 0.63 nM T86130 CGZ8W0 10152620 IC50 = 0.29 nM T86130 CC1F2P 10152817 IC50 = 6.6 nM T86130 CKE7G2 10153020 IC50 = 3.6 nM T86130 CJQ38N 10153070 IC50 = 0.6 nM T86130 C90YMF 10153095 IC50 = 350 nM T86130 CHC2U4 10161860 IC50 = 29 nM T86130 C9MZ6P 10162478 IC50 = 90 nM T86130 C27OAX 10164273 IC50 = 4.9 nM T86130 CCX2J0 10166459 IC50 = 107 nM T86130 CC4DS3 10174347 IC50 = 5.1 nM T86130 C6FEG3 10174365 IC50 = 1 nM T86130 CQ1G2F 10174690 IC50 = 0.5 nM T86130 CLR08U 10174895 IC50 = 0.21 nM T86130 CS49PU 10175357 IC50 = 0.8 nM T86130 C1I0RG 10175587 IC50 = 14 nM T86130 CJ1LW6 10179484 IC50 = 300 nM T86130 CA2D7Y 10179561 IC50 = 130 nM T86130 CAU46H 10179900 IC50 = 16 nM T86130 C41VQU 10180692 IC50 = 18 nM T86130 CT4NY2 10187032 IC50 = 3 nM T86130 CE5V8W 10187715 IC50 = 0.46 nM T86130 CS2JU4 10188054 IC50 = 1.1 nM T86130 CVGM95 10188056 IC50 = 0.77 nM T86130 CQ7R9N 10188398 IC50 = 56 nM T86130 CV01DN 10188683 IC50 = 0.67 nM T86130 C3ZVC5 10188879 IC50 = 4960 nM T86130 C96REN 10195992 IC50 = 1.1 nM T86130 C3DA8X 10196018 IC50 = 0.26 nM T86130 CGH38I 10196513 IC50 = 1.5 nM T86130 CYS7G2 10196582 IC50 = 2.4 nM T86130 CHT2O3 10196606 IC50 = 38 nM T86130 C9U4ZX 10196654 IC50 = 0.33 nM T86130 CM45IT 10196958 IC50 = 0.4 nM T86130 CQJ0O4 10202297 IC50 = 25 nM T86130 CGR6H4 10205401 IC50 = 81 nM T86130 CSJH35 10206665 IC50 = 0.19 nM T86130 C6OT2C 10207642 IC50 > 10000 nM T86130 CV9DG5 10208952 IC50 = 6740 nM T86130 CRH9F6 10210770 IC50 = 23 nM T86130 CLZW43 10211418 IC50 = 0.19 nM T86130 C6CZB1 10218171 IC50 = 7.8 nM T86130 CP5L4R 10218560 IC50 = 1.15 nM T86130 CS4D7N 10225908 IC50 = 180 nM T86130 CK8DC9 10229077 IC50 = 7 nM T86130 C2FGD4 10229869 IC50 = 20 nM T86130 CS69QU 10231058 IC50 = 0.09 nM T86130 CHB7A6 10231860 IC50 = 51 nM T86130 C1FH9Q 10232974 IC50 = 0.15 nM T86130 C8GN2D 10239567 IC50 = 8 nM T86130 CG31QV 10239586 IC50 = 0.46 nM T86130 C1W8UL 10239587 IC50 = 0.32 nM T86130 CRZY29 10239854 IC50 = 0.14 nM T86130 C4IP2F 10254400 IC50 = 20 nM T86130 CYE50Q 10255237 Ki = 2.512 nM T86130 CO82NU 10255795 IC50 = 0.5 nM T86130 CZ93JG 10255932 IC50 = 0.59 nM T86130 CH8QV9 10256855 IC50 = 0.26 nM T86130 CK01OV 10257083 IC50 = 0.37 nM T86130 C4WAR0 10257427 IC50 = 9.5 nM T86130 C5GEL4 10273950 IC50 = 582 nM T86130 C5LFE2 10277313 IC50 = 5.3 nM T86130 CDC2L7 10278812 IC50 = 10 nM T86130 CO7RI5 10280092 IC50 = 20 nM T86130 C7KA3Y 10280825 IC50 = 31 nM T86130 CTD53A 10281032 IC50 = 0.14 nM T86130 C4I3DN 10282143 IC50 = 0.1 nM T86130 C2YKU9 10282280 IC50 = 0.19 nM T86130 C25TMF 10282625 IC50 = 0.36 nM T86130 CC92ST 10299878 IC50 = 0.34 nM T86130 CV75FS 10300040 IC50 = 56 nM T86130 C7B2QP 10300477 IC50 = 296 nM T86130 CR0P9K 10300654 IC50 = 0.86 nM T86130 C1XO6Q 10301396 IC50 = 0.14 nM T86130 CRF0J3 10303859 IC50 = 26 nM T86130 CMDY64 10304716 IC50 = 0.13 nM T86130 CV5XW9 10311341 IC50 = 64 nM T86130 C3XSM2 10311568 IC50 = 3.4 nM T86130 C57XJE 10311889 IC50 = 1.1 nM T86130 CA5QX0 10311931 IC50 = 0.8 nM T86130 C58QCG 10312053 IC50 = 1.8 nM T86130 C8BY9F 10312159 IC50 = 8 nM T86130 CJ89QM 10312191 IC50 = 47 nM T86130 C1EF4L 10312394 IC50 = 40 nM T86130 C4K5NH 10324549 IC50 = 98 nM T86130 CIFT98 10325939 IC50 = 3 nM T86130 C2L1KB 10326465 IC50 = 30 nM T86130 C6GW8L 10345269 IC50 = 84 nM T86130 CY02JN 10364222 IC50 = 8000 nM T86130 C9FV3S 10371492 IC50 = 0.07 nM T86130 CT0KX3 10387865 IC50 = 0.9 nM T86130 C0RCX4 10388816 IC50 = 1.3 nM T86130 CB5WR2 10389159 IC50 = 46 nM T86130 CH67YI 10392222 IC50 = 2.2 nM T86130 C7ID9P 10393443 IC50 = 10 nM T86130 COG4R0 10394110 IC50 = 0.08 nM T86130 CG6U2D 10394204 IC50 = 0.1 nM T86130 C0IWH4 10413082 IC50 = 1 nM T86130 CF83CY 10431881 IC50 = 0.3 nM T86130 CE34WV 10458468 Ki = 1 nM T86130 CPO4V0 10458994 IC50 = 4.75 nM T86130 CEP1K2 10459011 IC50 = 12 nM T86130 CQR6B8 10460375 IC50 = 0.27 nM T86130 C4ZKT1 10460912 IC50 = 3.6 nM T86130 C0SA4N 10482036 IC50 = 0.5 nM T86130 CO3N2J 10483642 IC50 = 0.6 nM T86130 CV69GP 10484151 IC50 = 12 nM T86130 CWZ5V6 10504865 IC50 = 430 nM T86130 CSW56Y 10530953 IC50 = 250000 nM T86130 C9QPH4 10531085 IC50 = 250 nM T86130 C6HBM9 10533241 IC50 = 1200 nM T86130 CU2EI4 10553550 IC50 = 8 nM T86130 CJ9W1Y 10553946 IC50 = 6000 nM T86130 C7NA2C 10554760 IC50 = 5 nM T86130 C87YFN 10554892 IC50 = 54 nM T86130 C5Y0KP 10555697 IC50 = 1 nM T86130 CYP3A8 10555750 IC50 = 200 nM T86130 C59UDA 10555925 IC50 = 5 nM T86130 C0CL8F 10556023 IC50 = 40000 nM T86130 CT9ZW1 10556088 IC50 = 4 nM T86130 CKX96A 10556712 IC50 = 1 nM T86130 C8WJ2O 10578470 IC50 = 51000 nM T86130 CC9M7O 10601612 IC50 = 80000 nM T86130 CY4RD9 10601975 IC50 = 50000 nM T86130 CLZ3Y2 10602814 IC50 = 1500 nM T86130 CK3D5N 10602955 IC50 = 97 nM T86130 COK2J7 10603442 IC50 = 8 nM T86130 CNR14O 10603611 IC50 = 3 nM T86130 COP79I 10603612 IC50 = 400 nM T86130 CN8M6I 10604155 IC50 = 2 nM T86130 C4NB9D 10605027 IC50 = 2100 nM T86130 CL8S5A 10605189 IC50 = 9000 nM T86130 CW0G5F 10623968 IC50 = 1000 nM T86130 CGP3A4 10624203 IC50 = 2700 nM T86130 C0Z6TR 10625905 IC50 = 100 nM T86130 CP8L2Z 10627454 IC50 = 182000 nM T86130 C7BM5G 10627874 IC50 = 0.5 nM T86130 CHWG37 10628708 IC50 = 150 nM T86130 CZUJ51 10647467 IC50 = 350000 nM T86130 CM1WZ2 10649186 IC50 = 4200 nM T86130 C1QK7Z 10650919 IC50 = 3250 nM T86130 COJ16U 10651108 IC50 = 320 nM T86130 CBAP65 10651123 IC50 = 310 nM T86130 C7H0ZJ 10674294 IC50 = 3000 nM T86130 C6BV4N 10674312 IC50 = 22000 nM T86130 C63YSG 10674563 IC50 = 710 nM T86130 CCTS42 10675936 IC50 = 210 nM T86130 CJ7Q5V 10676968 IC50 = 20 nM T86130 C80JPK 10694497 IC50 = 5800 nM T86130 CCYV13 10695703 IC50 = 1000 nM T86130 CBK7W4 10696837 IC50 = 12000 nM T86130 CJ5TX0 10698275 IC50 = 34 nM T86130 CJ7I0X 10698961 IC50 = 140 nM T86130 C7WFD5 10699859 IC50 = 4 nM T86130 CFLS81 10699979 IC50 = 60 nM T86130 C63DSB 10700274 IC50 = 110 nM T86130 CF3U9R 10700352 IC50 = 30000 nM T86130 C71LVE 10718617 IC50 = 4200 nM T86130 C4ST0K 10721890 IC50 = 1100 nM T86130 C9F7KR 10722218 IC50 = 230 nM T86130 CIKA23 10743477 IC50 = 410 nM T86130 C7VB9P 10744975 IC50 = 18000 nM T86130 CTD0L4 10746264 IC50 = 20 nM T86130 C43UEP 10747979 IC50 = 15000 nM T86130 C96FOP 10769712 IC50 = 50000 nM T86130 CSX95N 10769729 IC50 = 3700 nM T86130 CZPU69 10793147 IC50 = 126000 nM T86130 C9TSD5 10793675 IC50 = 140 nM T86130 CZDB76 10793738 IC50 = 600 nM T86130 CZH78I 10793882 IC50 = 36000 nM T86130 C2H3WS 10794068 IC50 = 13 nM T86130 C3Y4KE 10795800 IC50 = 1 nM T86130 C45AQU 10815566 IC50 = 134 nM T86130 C2AQP4 10818386 IC50 = 3 nM T86130 CPA28R 10818515 IC50 = 250000 nM T86130 CNF06A 10838937 IC50 = 66000 nM T86130 C5HD8I 10838997 IC50 = 31 nM T86130 C0JUR8 10840473 IC50 = 14000 nM T86130 CUHR19 10841837 IC50 = 60000 nM T86130 CC0I1X 10916868 IC50 = 15000 nM T86130 C1CZ3O 10928862 IC50 = 67 nM T86130 CL7HW0 10960989 IC50 = 11400 nM T86130 CVBX27 10983911 IC50 = 800 nM T86130 CNWC78 11037638 IC50 = 2500 nM T86130 CV58GN 11037824 IC50 = 2300 nM T86130 C2A7GD 11123389 IC50 = 1200 nM T86130 CJQK52 11166204 IC50 = 790 nM T86130 CF0Q5M 11168346 IC50 = 310 nM T86130 CWE7R5 11168754 IC50 > 5000 nM T86130 CY12UD 11177161 IC50 > 5000 nM T86130 C3VA9H 11204176 IC50 = 150 nM T86130 C72DKJ 11212745 IC50 > 5000 nM T86130 CN17WU 11213435 IC50 > 5000 nM T86130 CHMU08 11214340 IC50 = 590 nM T86130 CAX6N8 11224267 IC50 > 5000 nM T86130 CJU14K 11249992 IC50 = 94 nM T86130 CU6JK8 11258559 IC50 = 1800 nM T86130 CM1OC4 11262030 IC50 = 0.25 nM T86130 CMJD76 11271230 IC50 > 5000 nM T86130 CGC54M 11272114 IC50 = 130 nM T86130 CT08ZV 11272553 IC50 = 480 nM T86130 C0GUA3 11296107 IC50 = 360 nM T86130 CA6EM9 11306407 IC50 > 5000 nM T86130 CZRP50 11337796 IC50 > 5000 nM T86130 COF9P4 11340507 IC50 = 31 nM T86130 CW09GY 11341120 IC50 = 300 nM T86130 CCB1I4 11341145 IC50 = 1300 nM T86130 CAV42L 11364489 IC50 = 790 nM T86130 C4R3UP 11376484 IC50 = 400 nM T86130 CQ3K4D 11385630 IC50 = 1200 nM T86130 C6BK8D 11387592 IC50 = 66 nM T86130 CY5B3Z 11408255 IC50 > 5000 nM T86130 C3MC5H 11441045 IC50 > 5000 nM T86130 C0C9IQ 11442204 IC50 > 1000 nM T86130 CW5CP6 11451270 IC50 > 5000 nM T86130 CXIM19 11454676 IC50 = 350 nM T86130 CC9Q5T 11478436 IC50 > 5000 nM T86130 CE43BF 11487182 IC50 = 1800 nM T86130 C78OKP 11495823 IC50 > 5000 nM T86130 C3U7CQ 11512183 IC50 = 3900 nM T86130 COK57Q 11513182 IC50 = 20 nM T86130 CAH69M 11547136 IC50 = 1000 nM T86130 C91BTP 11555311 IC50 = 280 nM T86130 CLOP01 11555715 IC50 = 150 nM T86130 CL1PB2 11568832 IC50 = 370 nM T86130 CR6GM5 11569874 IC50 = 790 nM T86130 CSQ4T0 11570705 IC50 = 1.7 nM T86130 C5SO0J 11577165 IC50 = 110 nM T86130 CX9YO2 11678416 IC50 = 520 nM T86130 COW1K8 11707191 IC50 = 19 nM T86130 CQ5IV6 11752188 IC50 = 170 nM T86130 C03NAR 11753632 IC50 = 4.7 nM T86130 CH6W5Y 11754265 IC50 = 0.2 nM T86130 C2YCH8 11758257 IC50 = 3 nM T86130 CT4D1K 11799915 IC50 = 18 nM T86130 C9LYZ4 11801761 IC50 = 1650 nM T86130 CZU3N7 11803206 IC50 = 40 nM T86130 C0Z8VB 11812359 IC50 = 2000 nM T86130 CUH0R5 11812936 IC50 = 58 nM T86130 CS24BW 11973730 IC50 = 2128 nM T86130 C0IWH9 12042474 IC50 = 18 nM T86130 CMD58G 12042475 IC50 = 20 nM T86130 CSV2F8 12042480 IC50 = 4500 nM T86130 CMV5Y6 12042481 IC50 = 640 nM T86130 CJ2T9L 12042482 IC50 = 870 nM T86130 CZS1A2 12043252 IC50 = 6.3 nM T86130 CR80BK 12114810 IC50 = 7300 nM T86130 CRKD02 12986829 IC50 = 80 nM T86130 C0ADG6 15541394 IC50 = 9460 nM T86130 C4TGS8 15984101 IC50 = 0.51 nM T86130 CMNW32 16041071 IC50 = 4.7 nM T86130 C3IO0P 16122691 IC50 = 3.4 nM T86130 CXI61L 16122692 IC50 = 1789.8 nM T86130 CGE4D6 16122706 IC50 = 1.6 nM T86130 C7SGL4 16122710 IC50 = 3.3 nM T86130 CNE2C4 16126658 Ki = 0.7943 nM T86130 CLDK13 16678632 IC50 = 822.9 nM T86130 CJF3Z9 16678636 IC50 = 18.5 nM T86130 CSKE71 16678739 IC50 = 1587.4 nM T86130 C9ZBU2 16678942 IC50 = 1.4 nM T86130 C3FZ4X 16678944 IC50 = 1054.4 nM T86130 CB3QP4 16679038 IC50 = 1.3 nM T86130 C9JW4X 16679039 IC50 = 2.3 nM T86130 CN64QM 16679040 IC50 = 2.8 nM T86130 C3C4EA 16679140 IC50 = 164.6 nM T86130 CJ8R3B 16679443 IC50 = 2019.7 nM T86130 CABL38 16679634 IC50 = 5832 nM T86130 CYVJ37 16679722 IC50 = 7.5 nM T86130 CG3FV0 16727128 IC50 = 0.3 nM T86130 C98SHM 17255620 IC50 > 1000000 nM T86130 C8EKT7 20599240 IC50 = 1.3 nM T86130 CBMW93 20599242 IC50 = 0.72 nM T86130 CRFH52 20599246 IC50 = 3 nM T86130 CQ8C7K 20599249 IC50 = 0.85 nM T86130 CGBP87 20687428 IC50 = 0.95 nM T86130 C9NHU3 20687429 IC50 = 0.46 nM T86130 CC3D1Z 20687430 IC50 = 0.13 nM T86130 CG9N6R 20687431 IC50 = 1.02 nM T86130 CE75LI 20687432 IC50 = 0.22 nM T86130 CJWR24 20687437 IC50 = 0.1 nM T86130 CCK1V3 20687440 IC50 = 0.1 nM T86130 C2UPQ9 20687441 IC50 = 0.36 nM T86130 C68ZCN 20687448 IC50 = 0.39 nM T86130 C6QU4T 20687449 IC50 = 0.4 nM T86130 C4WF5H 20687453 IC50 = 0.9 nM T86130 C2CQ7N 20687454 IC50 = 1.53 nM T86130 CTMN05 20687515 IC50 = 0.09 nM T86130 C2PZE7 20687518 IC50 = 0.33 nM T86130 CZ6MF7 20687535 IC50 = 11 nM T86130 C70LZV 20737909 IC50 = 2.9 nM T86130 C80IDM 20737927 IC50 = 4.4 nM T86130 C6QJW9 20737953 IC50 = 1.6 nM T86130 CK7AB3 20737962 IC50 = 13 nM T86130 C29ZYU 20793886 IC50 = 0.99 nM T86130 C8NLS0 20793887 IC50 = 0.5 nM T86130 C3DLN4 20793889 IC50 = 0.86 nM T86130 C4JB5Z 20793890 IC50 = 0.92 nM T86130 C2B7IK 20793891 IC50 = 0.85 nM T86130 C3BM8N 20793892 IC50 = 0.79 nM T86130 CY4E7U 20793893 IC50 = 0.3 nM T86130 CX0JL1 20793894 IC50 = 0.67 nM T86130 C4NJ2L 20793895 IC50 = 0.73 nM T86130 C1WN0S 20793908 IC50 = 0.28 nM T86130 C2D1UO 20793909 IC50 = 0.26 nM T86130 C1ZI3P 20793912 IC50 = 0.45 nM T86130 C27UDN 20793913 IC50 = 0.26 nM T86130 CVA8H3 20793914 IC50 = 0.22 nM T86130 CK0H4D 20793915 IC50 = 0.37 nM T86130 C3FW9R 20793916 IC50 = 1.11 nM T86130 C3W2BH 20793918 IC50 = 0.21 nM T86130 CF7TP9 20794038 IC50 = 0.21 nM T86130 CNG3Y6 20828691 IC50 = 0.03 nM T86130 CY56IV 21349552 IC50 = 560 nM T86130 C21CKN 22093322 IC50 = 3.9 nM T86130 C4SW7C 22093367 IC50 = 36 nM T86130 C67XLD 23562835 IC50 = 25 nM T86130 C0PZC6 23562840 IC50 = 2300 nM T86130 CAVY89 23636144 IC50 = 1966 nM T86130 C1VUH4 23636254 IC50 = 637 nM T86130 C6LR7V 23636255 IC50 = 4334 nM T86130 C5MSF6 23636502 IC50 = 770 nM T86130 C8RUT0 23647506 Ki = 1 nM T86130 CY48DN 23647507 Ki = 25.12 nM T86130 C5ZOX0 23647511 Ki = 19.95 nM T86130 C05OSP 23647512 Ki = 1.995 nM T86130 C0EIQ6 23647513 Ki = 2.512 nM T86130 CF5NL7 23647514 Ki = 251.19 nM T86130 CSE17D 23647515 Ki = 501.19 nM T86130 C8W3VT 23647516 Ki < 100000 nM T86130 C8U5OW 23647517 Ki < 1000 nM T86130 CXY98C 23647518 Ki = 25.12 nM T86130 CB81WR 23647519 Ki < 1000 nM T86130 C87BOW 23647520 Ki < 1000 nM T86130 CD8I5Y 23647521 Ki = 398.11 nM T86130 CLS32R 23647522 Ki = 251.19 nM T86130 CBZ31U 23647523 Ki = 63.1 nM T86130 C9LCX8 23647524 Ki = 0.7943 nM T86130 CX1YM3 23647538 IC50 = 36 nM T86130 CE8YM4 23647660 Ki = 1.585 nM T86130 C2MG7V 23647661 Ki = 316.23 nM T86130 C20ZAN 23647662 Ki = 6.31 nM T86130 CR93WK 23647663 Ki = 5.012 nM T86130 CE5U4G 23647664 Ki = 6.31 nM T86130 C1UH8Y 23647665 Ki = 25.12 nM T86130 CF6QZ5 23647666 Ki = 25.12 nM T86130 CJKQ21 23647667 Ki = 7.943 nM T86130 CRA49K 23647668 Ki = 1.995 nM T86130 CXZ84V 23647669 Ki = 1 nM T86130 C4RB9Q 23647670 Ki = 0.7943 nM T86130 CF9C7A 23647674 Ki = 2.512 nM T86130 CH5OS4 23647675 Ki = 1 nM T86130 CK40MN 23648174 IC50 = 0.305 nM T86130 CVF32G 24748310 IC50 = 15.5 nM T86130 CR9EP2 24748311 IC50 = 22.5 nM T86130 C9NAX1 24748312 IC50 = 26.8 nM T86130 CE7P6Q 24748313 IC50 = 18565.9 nM T86130 C7UX2P 24748314 IC50 = 22.7 nM T86130 CFA81R 24752916 IC50 = 0.0525 nM T86130 C2MER9 24986401 IC50 = 71 nM T86130 C2DNL6 24986402 IC50 = 18 nM T86130 C04GVM 24986403 IC50 = 10 nM T86130 C27WVS 24986404 IC50 = 2 nM T86130 CF9R2C 24986405 IC50 = 14 nM T86130 CTN6K7 24986762 IC50 = 8 nM T86130 CV8W1N 24986763 IC50 = 3 nM T86130 CI9YO4 24986765 IC50 = 3 nM T86130 CAR4B0 24986766 IC50 = 9 nM T86130 CPX9T4 24987117 IC50 = 83 nM T86130 CHV0E7 24987120 IC50 = 6 nM T86130 CT4PO2 24987475 IC50 = 22 nM T86130 C1ZB7M 24987477 IC50 = 46 nM T86130 C73QKH 24988955 IC50 = 11 nM T86130 C94AHE 24988956 IC50 = 3 nM T86130 CU5KQ0 24988957 IC50 = 2683 nM T86130 C06SLN 24988958 IC50 = 2 nM T86130 CIGA28 24989322 IC50 = 3 nM T86130 CH2J6T 24989709 IC50 = 8 nM T86130 C0IG5B 24990094 IC50 = 13 nM T86130 C60PZX 24990457 IC50 = 24 nM T86130 CQ3T8N 24990458 IC50 = 7 nM T86130 CPR03B 24990809 IC50 = 95 nM T86130 C7NZO5 24990811 IC50 = 22 nM T86130 CENO24 24990813 IC50 = 126 nM T86130 CMF95J 24991180 IC50 = 236 nM T86130 CG5FK3 24991181 IC50 = 19 nM T86130 CF9UL8 24991182 IC50 = 504 nM T86130 C02NZH 24991883 IC50 = 2 nM T86130 C0I5NG 24991884 IC50 = 9 nM T86130 CIF4D2 24991885 IC50 = 570 nM T86130 C5DCI0 24991886 IC50 = 11 nM T86130 CS98GW 25242385 IC50 = 45 nM T86130 C3J7GQ 28510125 EC50 = 10 nM T86130 CLX6T9 28510811 IC50 > 1000 nM T86130 CX5MP7 44232495 IC50 = 0.03 nM T86130 C8C7QA 44266063 IC50 = 0.9 nM T86130 C0YG4B 44266065 IC50 = 0.6 nM T86130 CCKZ78 44266073 IC50 = 0.5 nM T86130 C3DUE2 44266083 IC50 = 0.5 nM T86130 CV67IM 44266084 IC50 = 5.7 nM T86130 C9M1ZI 44266087 IC50 = 1.5 nM T86130 C4UAI1 44266091 IC50 = 1 nM T86130 CFK15X 44266103 IC50 = 67 nM T86130 CXMB30 44266106 IC50 = 0.4 nM T86130 C1CIU0 44266107 IC50 = 1 nM T86130 C0CTO3 44266115 IC50 = 1 nM T86130 CI6U4X 44266118 IC50 = 50 nM T86130 C5DZ3V 44266123 IC50 = 90 nM T86130 C47AWZ 44266143 IC50 = 0.5 nM T86130 C7PBY9 44266146 IC50 = 2.6 nM T86130 C4LP3V 44266154 IC50 = 40 nM T86130 C09PKF 44266158 IC50 = 180 nM T86130 CFE6C7 44266162 IC50 = 1.2 nM T86130 C5G6NA 44266166 IC50 = 9 nM T86130 CJGD42 44266167 IC50 = 6.7 nM T86130 CY24UK 44266169 IC50 = 6.9 nM T86130 CCY2Z7 44266171 IC50 = 0.2 nM T86130 CRI4H9 44266173 IC50 = 8.4 nM T86130 CC7S5G 44266174 IC50 = 0.4 nM T86130 C6TMV9 44266179 IC50 = 0.2 nM T86130 CKX9O1 44266184 IC50 = 0.3 nM T86130 C9AHY6 44266195 IC50 = 0.5 nM T86130 C2QVH0 44266204 IC50 = 1 nM T86130 C9X4CD 44266212 IC50 = 3.7 nM T86130 C5NI9F 44266217 IC50 = 1.2 nM T86130 CY8S0D 44266256 IC50 = 845 nM T86130 CML45U 44266270 IC50 = 3.5 nM T86130 CW26OR 44266277 IC50 = 0.5 nM T86130 CWQ3H6 44277247 IC50 = 0.1 nM T86130 CLD1E0 44277294 IC50 = 13 nM T86130 CIX4M7 44277304 IC50 = 0.1 nM T86130 C8HYQ2 44277327 IC50 = 0.3 nM T86130 CMN12S 44277340 IC50 = 6 nM T86130 CU4DX9 44277352 IC50 = 0.2 nM T86130 CL56IM 44277354 IC50 = 0.42 nM T86130 CA08RU 44277355 IC50 = 0.39 nM T86130 CSG1N6 44277413 IC50 = 8.2 nM T86130 CW1Z0Q 44278758 IC50 = 550 nM T86130 C7T3KB 44278759 IC50 = 4 nM T86130 C2KV8J 44278795 IC50 = 27 nM T86130 CV2KH0 44278903 IC50 = 2200 nM T86130 C5I7SD 44278996 IC50 = 120 nM T86130 C5EK4J 44278999 IC50 = 0.37 nM T86130 CXWO75 44279016 IC50 = 320 nM T86130 C4C7AF 44279040 IC50 = 240 nM T86130 CB4WJ6 44279041 IC50 = 12 nM T86130 C5VNO3 44279068 IC50 = 5500 nM T86130 COJ90U 44279069 IC50 = 61 nM T86130 C17FPH 44279070 IC50 = 57 nM T86130 CH6ES5 44279071 IC50 = 73 nM T86130 CWD41L 44279072 IC50 = 60 nM T86130 CXMO86 44279081 IC50 = 6.5 nM T86130 C8FW6I 44280570 IC50 = 2.7 nM T86130 CBG5C3 44283784 IC50 = 1.3 nM T86130 CG65HE 44283797 IC50 = 4.9 nM T86130 C3T4EO 44283971 IC50 = 0.88 nM T86130 C7CD9J 44283972 IC50 = 19.3 nM T86130 CTA6I7 44283985 IC50 = 2.1 nM T86130 CQC3T6 44284016 IC50 = 63 nM T86130 C5AG4M 44284069 IC50 = 4.1 nM T86130 C6N8CB 44284070 IC50 = 2.4 nM T86130 C27DZS 44284080 IC50 = 12.9 nM T86130 C1FM8B 44284102 IC50 = 1.7 nM T86130 CFP48W 44284103 IC50 = 2.8 nM T86130 CS47GU 44284171 IC50 = 1.56 nM T86130 CPH54Y 44284172 IC50 = 2.12 nM T86130 CO7Y3D 44284173 IC50 = 0.7 nM T86130 C0TC8Z 44284200 IC50 = 0.48 nM T86130 CZG56T 44284214 IC50 = 255 nM T86130 C6PW2K 44284215 IC50 = 1.15 nM T86130 CZI34O 44284227 IC50 = 0.7 nM T86130 CT0G2Q 44284229 IC50 = 0.92 nM T86130 CA48YS 44284230 IC50 = 0.23 nM T86130 CJ81ET 44284231 IC50 = 0.47 nM T86130 CT6C3W 44284239 IC50 = 4.09 nM T86130 CP4Y8X 44284243 IC50 = 23.15 nM T86130 CJB6G3 44284252 IC50 = 3.62 nM T86130 CQ13GI 44284315 IC50 = 1.48 nM T86130 C0WH4U 44284316 IC50 = 5.31 nM T86130 CN0R8X 44284320 IC50 = 1 nM T86130 C6QJ8L 44284386 IC50 = 0.7 nM T86130 CSLM73 44284387 IC50 = 4.3 nM T86130 CZHQ16 44284392 IC50 = 0.54 nM T86130 C5S8QO 44284406 IC50 = 4.06 nM T86130 CWF83Z 44284417 IC50 = 1.8 nM T86130 CIQP20 44284419 IC50 = 4.65 nM T86130 C8BR4A 44284432 IC50 = 2.6 nM T86130 C52WLJ 44284486 IC50 = 3.4 nM T86130 C9SL1V 44284494 IC50 = 9.18 nM T86130 CMZ5O4 44284517 IC50 = 16.3 nM T86130 CI1PJ9 44284534 IC50 = 0.35 nM T86130 C9D4ON 44284536 IC50 = 2.2 nM T86130 CI29RA 44284552 IC50 = 19.5 nM T86130 C5KNA7 44284553 IC50 = 4.62 nM T86130 CR7T5I 44284566 IC50 = 0.62 nM T86130 C28RWG 44284602 IC50 = 6.18 nM T86130 C6E7CQ 44284627 IC50 = 0.67 nM T86130 CH7S9Z 44284643 IC50 = 1.33 nM T86130 CS8M0W 44284678 IC50 = 0.31 nM T86130 C7FD8O 44287212 IC50 = 10 nM T86130 CMI31G 44287213 IC50 = 30 nM T86130 C8Q2BN 44287232 IC50 = 4 nM T86130 CP8TC0 44287259 IC50 = 1500 nM T86130 CQ4HY3 44287263 IC50 = 4600 nM T86130 CZ14NO 44287314 IC50 = 6 nM T86130 C05PBG 44287325 IC50 = 7 nM T86130 CC7FU2 44287361 IC50 = 4 nM T86130 CB3QL0 44287366 IC50 = 430 nM T86130 C8PNW6 44287371 IC50 = 25 nM T86130 CHVX89 44287372 IC50 = 80 nM T86130 CG89OU 44287374 IC50 = 1400 nM T86130 CIYW63 44287376 IC50 = 30 nM T86130 CGP0R6 44287377 IC50 = 30 nM T86130 CKR81O 44287421 IC50 = 660 nM T86130 C1CY7D 44287437 IC50 = 2 nM T86130 CRYH51 44287450 IC50 = 50 nM T86130 CT7D3A 44287492 IC50 = 2 nM T86130 CQ53HZ 44287494 IC50 = 14 nM T86130 C5RAT7 44287495 IC50 = 320 nM T86130 CF92QD 44287496 IC50 = 25 nM T86130 C3TX1W 44287512 IC50 = 1500 nM T86130 CX58EV 44287520 IC50 = 16 nM T86130 CWD41T 44287525 IC50 = 5500 nM T86130 CS7V1M 44287597 IC50 = 3400 nM T86130 CQ0SM2 44287598 IC50 = 1600 nM T86130 C4B0KC 44287626 IC50 = 4 nM T86130 CC7Z0M 44287661 IC50 = 410 nM T86130 C02VME 44287662 IC50 = 50 nM T86130 CO7WI9 44287663 IC50 = 260 nM T86130 CJ7D1I 44287679 IC50 = 6 nM T86130 CBA7C4 44287692 IC50 = 520 nM T86130 CKED14 44287693 IC50 = 1620 nM T86130 C8SIC1 44287702 IC50 = 40 nM T86130 CI21KO 44287704 IC50 = 45 nM T86130 CKJL31 44287727 IC50 = 60 nM T86130 CLZS95 44287743 IC50 = 50 nM T86130 CU31NV 44288627 IC50 = 0.13 nM T86130 CI2C3Y 44288628 IC50 = 0.25 nM T86130 CQ48WG 44288629 IC50 = 0.22 nM T86130 CQG2B8 44288785 IC50 = 0.13 nM T86130 CT0N2E 44288793 IC50 = 1.79 nM T86130 CV9Y2B 44288796 IC50 = 0.5 nM T86130 CAU49W 44288817 IC50 = 0.19 nM T86130 C6WKT1 44288845 IC50 = 0.17 nM T86130 C0BQ5O 44288950 IC50 = 0.18 nM T86130 C4XLV9 44289093 IC50 = 0.41 nM T86130 CDK92F 44289115 IC50 = 3.65 nM T86130 CDX08U 44291565 IC50 = 2400 nM T86130 CK9L6N 44299090 IC50 = 0.36 nM T86130 CH3Z2J 44299091 IC50 = 0.16 nM T86130 C1E8PU 44299097 IC50 = 0.21 nM T86130 C09OHT 44299108 IC50 = 0.1 nM T86130 CDVQ24 44299109 IC50 = 0.1 nM T86130 CTL1J5 44299112 IC50 = 0.11 nM T86130 C9F0HG 44299113 IC50 = 0.14 nM T86130 CXS1I7 44299114 IC50 = 0.25 nM T86130 CNDW49 44299159 IC50 = 0.08 nM T86130 CCT6K8 44299160 IC50 = 0.1 nM T86130 C9IGM3 44299178 IC50 = 0.13 nM T86130 C1JO5I 44307818 IC50 = 36.8 nM T86130 CE7LC4 44309967 IC50 = 0.41 nM T86130 C9HJ0O 44309968 IC50 = 1.9 nM T86130 CY6S2Q 44309985 IC50 = 1.1 nM T86130 CA8I7F 44309987 IC50 = 0.05 nM T86130 C6T4NH 44310021 IC50 = 0.73 nM T86130 C6B7YP 44310233 IC50 = 0.11 nM T86130 C5BGH0 44310255 IC50 = 0.37 nM T86130 C9BE3Y 44310286 IC50 = 0.61 nM T86130 C30PME 44310537 IC50 = 0.34 nM T86130 C9VOA3 44310538 IC50 = 1.1 nM T86130 CJEU74 44310553 IC50 = 3.2 nM T86130 CL8E2H 44310557 IC50 = 0.17 nM T86130 C9RQB2 44313545 IC50 > 100000 nM T86130 C2TLH6 44313669 IC50 >> 100000 nM T86130 C4JO7L 44314429 IC50 = 0.69 nM T86130 CBN9O7 44314430 IC50 = 0.54 nM T86130 CIW4N3 44314551 IC50 = 1.7 nM T86130 CF34ZY 44314636 IC50 = 0.79 nM T86130 C8XGA3 44314668 IC50 = 140 nM T86130 C9ABU8 44314711 IC50 = 0.27 nM T86130 C7DY6K 44317611 IC50 = 2.6 nM T86130 CZU6R4 44321165 IC50 = 20 nM T86130 CPXY32 44321347 IC50 = 2.6 nM T86130 C7NHZ0 44321348 IC50 = 8 nM T86130 C4FZ3B 44321429 IC50 = 800 nM T86130 CA90JV 44321433 IC50 = 9.8 nM T86130 CV2TQ6 44321444 IC50 = 800 nM T86130 CIA81W 44321445 IC50 = 2400 nM T86130 CD8ZP9 44321513 IC50 = 1800 nM T86130 C8VTY4 44321530 IC50 = 3 nM T86130 C9V5DG 44324292 IC50 = 0.23 nM T86130 CYE8B9 44324396 IC50 = 0.38 nM T86130 CI1PA9 44324431 IC50 = 10 nM T86130 C5TSO8 44324472 IC50 = 0.15 nM T86130 CW4K2Z 44324473 IC50 = 0.65 nM T86130 C7H1TW 44324487 IC50 = 0.5 nM T86130 C2ULQ5 44324488 IC50 = 0.28 nM T86130 CP2B8I 44324517 IC50 = 0.16 nM T86130 C5GF7J 44324561 IC50 = 0.14 nM T86130 C27DSJ 44324581 IC50 = 1.43 nM T86130 C7ROW6 44324587 IC50 = 0.15 nM T86130 CXG2Y7 44324588 IC50 = 0.54 nM T86130 CO2FS0 44324632 IC50 = 7 nM T86130 CX9DS5 44324688 IC50 = 0.52 nM T86130 CQ4H6L 44324703 IC50 = 360 nM T86130 C7R5ZM 44324730 IC50 = 4.5 nM T86130 CMS19Y 44324731 IC50 = 0.22 nM T86130 C3TQ9H 44324732 IC50 = 0.14 nM T86130 CKY7S0 44324733 IC50 = 257 nM T86130 CW2G4X 44324735 IC50 = 1.01 nM T86130 CQ53DR 44324768 IC50 = 0.52 nM T86130 C50RSE 44324774 IC50 = 1.33 nM T86130 C16XST 44324776 IC50 = 0.35 nM T86130 C4NK8T 44324794 IC50 = 0.24 nM T86130 C03KOG 44324807 IC50 = 0.11 nM T86130 CFAV34 44324809 IC50 = 0.09 nM T86130 CWG84B 44324812 IC50 = 1.12 nM T86130 CJN8B3 44324819 IC50 = 2.4 nM T86130 C2OJI4 44324820 IC50 = 0.92 nM T86130 COIG83 44324854 IC50 = 192 nM T86130 C3C9RN 44324855 IC50 = 0.53 nM T86130 COF9V0 44324856 IC50 = 45 nM T86130 CE3TH4 44330475 IC50 = 25.3 nM T86130 CL6RA9 44330517 IC50 = 48 nM T86130 CBME25 44330518 IC50 = 237 nM T86130 C4BJK6 44330548 IC50 = 82.1 nM T86130 CN0S7M 44330565 IC50 = 61.3 nM T86130 CA3UX5 44330581 IC50 = 25 nM T86130 C13PBU 44330595 IC50 = 9.3 nM T86130 CXTA89 44330626 IC50 = 16.8 nM T86130 CWN4L8 44330629 IC50 = 1.1 nM T86130 CJ4E6H 44330660 IC50 = 51.1 nM T86130 C94KJY 44331292 IC50 = 20 nM T86130 C4U3AT 44331317 IC50 = 2900 nM T86130 CC0WY4 44331360 IC50 = 262000 nM T86130 C28LKV 44331361 IC50 = 75000 nM T86130 C9OR1E 44331370 IC50 = 37000 nM T86130 C38KEV 44331371 IC50 = 247000 nM T86130 C9ZX3P 44331372 IC50 = 6400 nM T86130 CAX0Q1 44331387 IC50 = 45 nM T86130 CE05GV 44331388 IC50 = 103000 nM T86130 C3PKO5 44331392 IC50 = 16.5 nM T86130 CR9Y6C 44331393 IC50 = 5900 nM T86130 C57MOC 44331437 IC50 = 7300 nM T86130 CIE52Q 44331438 IC50 > 500000 nM T86130 CLO50N 44331464 IC50 = 11000 nM T86130 CILD16 44331474 IC50 = 29 nM T86130 C8S7IB 44331476 IC50 = 98 nM T86130 CRJM13 44331480 IC50 = 3 nM T86130 C18MVS 44332140 IC50 = 0.6 nM T86130 C0I5FT 44332251 IC50 = 20000 nM T86130 CY4B7J 44332254 IC50 = 3000 nM T86130 CW92LG 44341672 IC50 = 100 nM T86130 CPLZ63 44341717 IC50 = 420 nM T86130 C4ZHY3 44341719 IC50 = 23 nM T86130 C0Z4MP 44341727 IC50 = 300 nM T86130 CK3NF7 44341748 IC50 = 76 nM T86130 CE48RA 44341766 IC50 = 40 nM T86130 CFGS32 44341894 IC50 = 115000 nM T86130 CX46NY 44343237 IC50 = 1100 nM T86130 CF38BE 44343238 IC50 = 8300 nM T86130 CFQ6R5 44343239 IC50 = 8800 nM T86130 C8L4HI 44343263 IC50 = 3800 nM T86130 CU5Z9G 44343282 IC50 = 3200 nM T86130 C6AJ8U 44343283 IC50 = 1200 nM T86130 C80DNY 44343284 IC50 = 7400 nM T86130 C5A0BF 44343310 IC50 = 4200 nM T86130 CHP40V 44343311 IC50 = 11800 nM T86130 CFX5B7 44343326 IC50 > 100000 nM T86130 CNMQ48 44343327 IC50 = 3600 nM T86130 C9E8NP 44343328 IC50 = 2800 nM T86130 CV9M6T 44343453 IC50 = 8600 nM T86130 CL8E3T 44343454 IC50 = 50 nM T86130 COM1C6 44343455 IC50 = 9 nM T86130 CQ8Z1H 44343585 IC50 = 4200 nM T86130 CU0A2D 44343587 IC50 = 37000 nM T86130 CW97VR 44343589 IC50 = 13000 nM T86130 CHX5I8 44343599 IC50 = 2200 nM T86130 C53TVL 44343600 IC50 = 400 nM T86130 CHF18Y 44343602 IC50 > 100000 nM T86130 C0LGN6 44343603 IC50 = 59000 nM T86130 CO12WD 44343604 IC50 = 25000 nM T86130 CO7R5Y 44343621 IC50 > 100000 nM T86130 C35FPB 44343634 IC50 = 14000 nM T86130 C19TDW 44343641 IC50 = 1500 nM T86130 CPZE98 44343642 IC50 = 40000 nM T86130 CJ73KU 44343656 IC50 = 3000 nM T86130 CHQ96V 44343657 IC50 = 88000 nM T86130 C6K8DG 44343677 IC50 = 60000 nM T86130 CC35LO 44343703 IC50 = 800 nM T86130 C0I9YS 44343704 IC50 = 1100 nM T86130 CRUH62 44343705 IC50 = 160 nM T86130 C7KBF2 44350523 IC50 = 2 nM T86130 C5RY0Q 44350524 IC50 = 2 nM T86130 CWAE26 44350531 IC50 = 1 nM T86130 CJ3I6U 44350550 IC50 = 180 nM T86130 C4WE3Z 44350592 IC50 = 1.5 nM T86130 CLMC54 44350593 IC50 = 0.8 nM T86130 C9J7RQ 44350598 IC50 = 0.7 nM T86130 CE73CR 44350599 IC50 = 2 nM T86130 CJM01Q 44351896 IC50 = 0.52 nM T86130 C0IM6J 44351897 IC50 = 4.3 nM T86130 C6YO5K 44352017 IC50 = 184 nM T86130 C3O0BZ 44352053 IC50 = 16 nM T86130 C8KX5D 44352063 IC50 = 2.7 nM T86130 CP3J0A 44352167 IC50 = 0.54 nM T86130 C6H8EV 44370061 IC50 = 69 nM T86130 C2CIL9 44370062 IC50 = 11 nM T86130 CHON83 44370159 IC50 = 12 nM T86130 CF7V2B 44370160 IC50 = 18 nM T86130 CN4DX6 44370168 IC50 = 150 nM T86130 CJK9Q2 44370249 IC50 = 81 nM T86130 CX3L1Z 44370279 IC50 = 900 nM T86130 CTM71W 44370296 IC50 = 105 nM T86130 C0M4DW 44370366 IC50 = 45 nM T86130 C3LYR9 44370367 IC50 = 1100 nM T86130 COE0F8 44370368 IC50 = 1600 nM T86130 COAZ63 44370391 IC50 = 30 nM T86130 CQ8X0O 44370392 IC50 = 1600 nM T86130 C3LNK4 44370407 IC50 = 51 nM T86130 CRK8J6 44370788 IC50 = 3 nM T86130 CY54XC 44370792 IC50 = 1.4 nM T86130 C3XLQ5 44370799 IC50 = 26 nM T86130 C9M7YU 44370805 IC50 = 2.6 nM T86130 CQ51NH 44370853 IC50 = 13 nM T86130 CSTG72 44370868 IC50 = 544 nM T86130 CZ36HU 44370874 IC50 = 1500 nM T86130 C7HT3X 44370875 IC50 = 362 nM T86130 CB7AP3 44370903 IC50 = 3.1 nM T86130 CLVB32 44370911 IC50 = 0.31 nM T86130 C1SBF8 44370923 IC50 = 0.53 nM T86130 C7W9ZP 44370948 IC50 = 0.74 nM T86130 CR4IH9 44370977 IC50 = 11 nM T86130 CSYT51 44370978 IC50 = 2.1 nM T86130 C0QVA6 44370979 IC50 = 0.55 nM T86130 C94PNA 44371011 IC50 = 22 nM T86130 C4H3GE 44371047 IC50 = 8.9 nM T86130 CM9I6N 44371105 IC50 = 3.2 nM T86130 CKN9P4 44371123 IC50 = 1.5 nM T86130 CT4M5B 44371219 IC50 = 0.5 nM T86130 C4Z6UP 44371960 IC50 = 1.1 nM T86130 C41IKQ 44372067 IC50 = 3.9 nM T86130 C6JO8A 44372076 IC50 = 0.86 nM T86130 CFAL73 44372087 IC50 = 1.31 nM T86130 CE7TW6 44372098 IC50 = 0.44 nM T86130 C05OBK 44372138 IC50 = 2.3 nM T86130 C9H4VF 44372139 IC50 = 1.7 nM T86130 CN6QA9 44372166 IC50 = 1.7 nM T86130 CR9UF7 44372194 IC50 = 1.8 nM T86130 C4PM2U 44372195 IC50 = 3.2 nM T86130 CUYR80 44372206 IC50 = 3.8 nM T86130 C7I1RY 44372215 IC50 = 4.77 nM T86130 C9GP4S 44372251 IC50 = 1.88 nM T86130 CYTI54 44372263 IC50 = 0.67 nM T86130 C2XC8M 44372264 IC50 = 0.48 nM T86130 CR72AK 44372286 IC50 = 1.3 nM T86130 COSR59 44372318 IC50 = 2055 nM T86130 CE6N2I 44372331 IC50 = 152 nM T86130 CBAO19 44372332 IC50 = 28450 nM T86130 C1Z7CY 44372341 IC50 = 1.61 nM T86130 C4UJW3 44372342 IC50 = 0.92 nM T86130 C8ZQ0L 44372361 IC50 = 26.5 nM T86130 CEQ75T 44372434 IC50 = 3.6 nM T86130 CSI3C0 44372487 IC50 = 1.6 nM T86130 CM7ZH6 44372501 IC50 = 0.9 nM T86130 CH7S6U 44376211 IC50 = 3190 nM T86130 CH4MU3 44376214 IC50 = 60 nM T86130 CRE1B4 44376217 IC50 = 317 nM T86130 C5KVB3 44376224 IC50 = 4180 nM T86130 C2R4TX 44376231 IC50 = 245 nM T86130 CC52VL 44376237 IC50 = 170 nM T86130 CMD62U 44376238 IC50 = 3550 nM T86130 CEF42D 44376239 IC50 = 0.74 nM T86130 CFW36E 44376240 IC50 = 0.87 nM T86130 CK47CU 44376243 IC50 = 6490 nM T86130 CW0H8C 44376261 IC50 = 8870 nM T86130 C8GY5J 44376266 IC50 = 42500 nM T86130 CC8Z4M 44376271 IC50 = 4360 nM T86130 CDS4G0 44376294 IC50 = 0.75 nM T86130 C5BSI8 44376295 IC50 = 1.1 nM T86130 CWIN53 44376301 IC50 = 74 nM T86130 C8AD4T 44376320 IC50 = 152 nM T86130 CH5GD2 44376330 IC50 = 1060 nM T86130 CWYC71 44376340 IC50 = 0.37 nM T86130 C2WGQ4 44376341 IC50 = 0.82 nM T86130 C6K8NC 44376358 IC50 = 0.88 nM T86130 C46TDI 44376359 IC50 = 1.4 nM T86130 C8L1TK 44376406 IC50 = 4.6 nM T86130 C6PVS9 44376433 IC50 = 3.6 nM T86130 C97ZAK 44376448 IC50 = 187 nM T86130 CQDL60 44376471 IC50 = 135 nM T86130 C9HN6X 44376473 IC50 = 4200 nM T86130 CA5FL8 44376490 IC50 = 210 nM T86130 CSQ69H 44376497 IC50 = 38 nM T86130 C5KMG8 44376499 IC50 = 220 nM T86130 CZVT14 44376500 IC50 = 160 nM T86130 C0YO6I 44376511 IC50 = 230 nM T86130 C5MAV7 44376535 IC50 = 610 nM T86130 CD14GJ 44376536 IC50 = 23 nM T86130 C89DHB 44376537 IC50 = 32 nM T86130 C08ENQ 44376538 IC50 = 127 nM T86130 CZP1U5 44376543 IC50 = 5250 nM T86130 CR1B9X 44376546 IC50 = 53 nM T86130 CVG9A7 44376558 IC50 = 90 nM T86130 C8MFX6 44376564 IC50 = 12 nM T86130 C52WNX 44376570 IC50 = 1.2 nM T86130 C4W8FE 44376577 IC50 = 2.4 nM T86130 C3B5QU 44376590 IC50 = 2.4 nM T86130 CWUF18 44376595 IC50 = 4470 nM T86130 C3GOM9 44376596 IC50 = 820 nM T86130 C12VKX 44376615 IC50 = 4 nM T86130 C9UFJ0 44376618 IC50 = 17 nM T86130 CIS16K 44376619 IC50 = 5.3 nM T86130 CG7MJ3 44376633 IC50 = 20 nM T86130 CBQH15 44376636 IC50 = 320 nM T86130 CEJ73X 44376637 IC50 = 53 nM T86130 CAD81T 44376653 IC50 = 7000 nM T86130 CGK95E 44376672 IC50 = 590 nM T86130 C60POD 44376725 IC50 = 1000 nM T86130 CDR94J 44376726 IC50 = 59 nM T86130 CT8V2E 44376727 IC50 = 8.2 nM T86130 C3TW0O 44376733 IC50 = 3800 nM T86130 C2MZ9C 44376840 IC50 = 240 nM T86130 CQ6T1Z 44376859 IC50 = 97 nM T86130 CVLA70 44376877 IC50 = 91 nM T86130 CRN76F 44379557 IC50 = 140 nM T86130 CL5OD1 44379618 IC50 = 2 nM T86130 CZG4E6 44379629 IC50 = 2.7 nM T86130 CU94FN 44379630 IC50 = 14 nM T86130 CCK21Y 44379802 IC50 = 220 nM T86130 CR14MG 44379874 IC50 = 2200 nM T86130 C1WC3A 44379915 IC50 = 400 nM T86130 C9RVC8 44379927 IC50 = 60 nM T86130 C19WFZ 44379944 IC50 = 5 nM T86130 C02HZN 44379945 IC50 = 1500 nM T86130 CCY53E 44379967 IC50 = 7400 nM T86130 C2FR5H 44379985 IC50 = 2800 nM T86130 C1GDE4 44382099 IC50 = 1.5 nM T86130 CYX48W 44382102 IC50 = 28 nM T86130 C8UG4P 44382103 IC50 = 0.33 nM T86130 CG0XQ8 44382104 IC50 = 14 nM T86130 CDO7I6 44382111 IC50 = 0.53 nM T86130 C7A5EH 44382119 IC50 = 53 nM T86130 C4PV0Z 44382160 IC50 = 44 nM T86130 C93FHP 44382162 IC50 = 735 nM T86130 CY40TS 44382171 IC50 = 0.39 nM T86130 CK2GI4 44382174 IC50 = 1.1 nM T86130 C6MEZ0 44382232 IC50 = 0.47 nM T86130 C0WH5I 44382242 IC50 = 23 nM T86130 C5WE8L 44382283 IC50 = 28 nM T86130 C6AO0T 44382423 IC50 = 0.22 nM T86130 CY2C6E 44382469 IC50 = 0.37 nM T86130 CPSO78 44382497 IC50 = 0.1 nM T86130 CO5FU2 44382554 IC50 = 1.3 nM T86130 CNFM87 44382556 IC50 = 4.4 nM T86130 CIEX15 44382584 IC50 = 0.55 nM T86130 CQHD50 44382635 IC50 = 0.16 nM T86130 C0RL7W 44382645 IC50 = 680 nM T86130 CUC7Q0 44382647 IC50 = 275 nM T86130 C05FRE 44382649 IC50 = 0.17 nM T86130 CGMN67 44382676 IC50 = 0.77 nM T86130 CUA54V 44382682 IC50 = 65 nM T86130 CAR47D 44382683 IC50 = 0.19 nM T86130 C28BMU 44382684 IC50 = 0.11 nM T86130 C0AY8L 44382685 IC50 = 0.97 nM T86130 CSB73O 44382695 IC50 = 81 nM T86130 CTCQ75 44382696 IC50 = 105 nM T86130 C45QUC 44382714 IC50 = 0.22 nM T86130 C6TLQ9 44382715 IC50 = 0.27 nM T86130 C91HRV 44382716 IC50 = 1.1 nM T86130 C1OP9Q 44382723 IC50 = 2.7 nM T86130 CS5L2W 44382724 IC50 = 45 nM T86130 C6I8BY 44382725 IC50 = 7 nM T86130 CLMI61 44382729 IC50 = 0.75 nM T86130 C2NC6F 44382730 IC50 = 150 nM T86130 CDK46W 44382769 IC50 = 15 nM T86130 CRL9V3 44382770 IC50 = 0.21 nM T86130 C0BR5U 44382771 IC50 = 1.2 nM T86130 C1QF5Y 44382777 IC50 = 0.07 nM T86130 CSIT45 44382810 IC50 = 1 nM T86130 C7L5TE 44382824 IC50 = 4.1 nM T86130 CL2G1B 44382830 IC50 = 1.2 nM T86130 CNG53Z 44385649 IC50 = 6 nM T86130 C35EGC 44385761 IC50 = 35250 nM T86130 C5O3XJ 44385762 IC50 = 263000 nM T86130 CZ64MK 44385829 IC50 = 310 nM T86130 CA3N4W 44385881 IC50 = 19520 nM T86130 CSK57E 44386199 IC50 = 90 nM T86130 CBED40 44386259 IC50 = 2 nM T86130 C4U1DB 44386260 IC50 = 3 nM T86130 CU70QC 44386462 IC50 = 425 nM T86130 C58NCI 44386643 IC50 = 280 nM T86130 CPI4O2 44386693 IC50 = 2340 nM T86130 CL9J3U 44386852 IC50 = 330 nM T86130 CO5G8S 44386853 IC50 = 41000 nM T86130 CD5U7L 44386854 IC50 = 5100 nM T86130 CF01PT 44386897 IC50 = 25200 nM T86130 CJR3W1 44386898 IC50 > 800000 nM T86130 CO9FC7 44386899 IC50 = 12 nM T86130 CJ31MT 44386900 IC50 = 170 nM T86130 CW1RG4 44386943 IC50 = 25 nM T86130 CP68GE 44386995 IC50 = 12 nM T86130 C40EDC 44387053 IC50 = 170 nM T86130 C2N0ZE 44387121 IC50 = 17 nM T86130 CCX6L5 44387126 IC50 = 4100 nM T86130 C5LE7N 44387143 IC50 = 47 nM T86130 CY47GD 44387170 IC50 = 15 nM T86130 CMW8I6 44387171 IC50 = 9 nM T86130 C9SQ6Y 44387471 IC50 = 0.38 nM T86130 CPF0C7 44391984 IC50 = 48 nM T86130 CJ0F4M 44392041 IC50 = 0.65 nM T86130 CN81YW 44392042 IC50 = 1.1 nM T86130 CRH2S8 44392056 IC50 = 54 nM T86130 C5Q0GB 44392059 IC50 = 0.4 nM T86130 C98BOG 44392077 IC50 = 3300 nM T86130 CF80BO 44392079 IC50 = 7100 nM T86130 CGCX94 44392080 IC50 = 4.9 nM T86130 C27PUA 44392081 IC50 = 23 nM T86130 CEZB63 44392089 IC50 = 1700 nM T86130 CA4I3V 44392090 IC50 = 5800 nM T86130 C8M1TZ 44392091 IC50 = 940 nM T86130 CCZP92 44392102 IC50 > 100000 nM T86130 CZ1QE6 44392107 IC50 = 650 nM T86130 CVL3M5 44392121 IC50 = 5000 nM T86130 C1KRF9 44392122 IC50 = 620 nM T86130 C1MAG8 44392127 IC50 = 1700 nM T86130 CMH3G8 44392128 IC50 = 3.1 nM T86130 CWYD48 44392129 IC50 = 3.8 nM T86130 CZ8Q3W 44392139 IC50 > 100000 nM T86130 C49PHZ 44392140 IC50 = 8.4 nM T86130 C6ES7P 44392141 IC50 = 16 nM T86130 C8PGE1 44392145 IC50 = 1700 nM T86130 C8UM6X 44392146 IC50 = 1100 nM T86130 CMZ9V5 44392152 IC50 = 930 nM T86130 C1X0JQ 44392158 IC50 = 11 nM T86130 CVL45M 44392163 IC50 = 7000 nM T86130 CGND62 44392164 IC50 = 5300 nM T86130 C26VSE 44392261 IC50 = 76 nM T86130 CE3DI8 44392264 IC50 = 10 nM T86130 CE25RK 44392270 IC50 = 295 nM T86130 CLQ8Y0 44392271 IC50 = 32 nM T86130 CGSL49 44392280 IC50 = 121 nM T86130 C91IQE 44392282 IC50 = 26 nM T86130 C9UO4Z 44392292 IC50 = 3.8 nM T86130 CAU2P5 44392298 IC50 = 148 nM T86130 CNZG37 44392303 IC50 = 20 nM T86130 C8PT2R 44392305 IC50 = 82 nM T86130 CMXJ94 44392349 IC50 = 1.6 nM T86130 CTWA32 44392356 IC50 = 7.1 nM T86130 CF68RZ 44392358 IC50 = 1.4 nM T86130 CB58ID 44392367 IC50 > 1000 nM T86130 CS8T3X 44392369 IC50 = 14 nM T86130 C7F2GI 44397691 IC50 = 6 nM T86130 C6BCF7 44397817 IC50 = 60 nM T86130 CMD53C 44397963 IC50 = 13 nM T86130 CBXI76 44397964 IC50 = 300 nM T86130 C7UD4M 44397965 IC50 = 10 nM T86130 CT07HC 44397966 IC50 = 11 nM T86130 CC6PQ8 44419294 Ki = 6.31 nM T86130 C49FEK 44419307 Ki = 5.012 nM T86130 C4U9VZ 44419310 Ki = 50.12 nM T86130 CK6XH7 44419338 Ki = 3.981 nM T86130 CX8GO2 44419339 Ki = 19.95 nM T86130 C4OAE7 44419343 Ki = 1.995 nM T86130 CSM92V 44430322 IC50 = 525 nM T86130 CVW46K 44430323 IC50 = 299 nM T86130 CWNG14 44430326 IC50 = 1597 nM T86130 CJ9H5K 44430327 IC50 = 54 nM T86130 C9YOZ7 44430328 IC50 = 657 nM T86130 CWT9L4 44430330 IC50 = 2740 nM T86130 CYPJ54 44430331 IC50 = 25600 nM T86130 C0C9KZ 44430332 IC50 = 462 nM T86130 CB1Y6P 44436334 IC50 = 0.0372 nM T86130 CCL8P7 44436335 IC50 = 185.6 nM T86130 CHV0B9 44436337 IC50 = 444 nM T86130 C1LO3N 44436338 IC50 = 340 nM T86130 CY0R6K 44436339 IC50 = 0.305 nM T86130 CX0GY5 44436341 IC50 = 344 nM T86130 CQT51V 44436342 IC50 = 419.5 nM T86130 C3CFA4 44436344 IC50 = 655 nM T86130 C9A8SD 44436345 IC50 = 27.5 nM T86130 CO4YE7 44454480 IC50 = 510 nM T86130 C1ZNQ8 44454481 IC50 = 2700 nM T86130 C3AGH7 44454515 IC50 > 5000 nM T86130 CI1A9S 44454544 IC50 = 520 nM T86130 C3IW1E 44454549 IC50 = 830 nM T86130 CDW2G9 44454578 IC50 = 1540 nM T86130 CS81QU 44454580 IC50 = 340 nM T86130 C72NXQ 44454604 IC50 = 460 nM T86130 CN2D6B 44454606 IC50 = 740 nM T86130 CFY48V 44454634 IC50 > 5000 nM T86130 CK5EN8 44454635 IC50 = 570 nM T86130 CW5SF4 44454656 IC50 = 3200 nM T86130 C5WF3A 44454658 IC50 = 2100 nM T86130 CIU9A7 44454686 IC50 > 5000 nM T86130 C5OZ7S 44454712 IC50 > 5000 nM T86130 CCPW89 44454736 IC50 = 730 nM T86130 CX0N7J 44454738 IC50 = 5 nM T86130 C43JVS 44461305 IC50 = 47 nM T86130 CAYL90 44461422 IC50 = 23 nM T86130 CNI07Z 44461423 IC50 = 2 nM T86130 C5LSI3 44461449 IC50 = 2 nM T86130 C5DYA0 44461450 IC50 = 200 nM T86130 CM92YQ 44461466 IC50 = 0.42 nM T86130 C5VZ2J 44461467 IC50 = 1.3 nM T86130 CQ27FH 44461495 IC50 = 0.49 nM T86130 CN4SE8 44461500 IC50 = 1.15 nM T86130 CA3L6Z 44461502 IC50 = 1.9 nM T86130 C67DER 44461523 IC50 = 0.47 nM T86130 CW7B5R 44461524 IC50 = 2.5 nM T86130 CDN8U3 44461547 IC50 = 1300 nM T86130 C6F2RG 44461564 IC50 = 33 nM T86130 C3T5GB 44461584 IC50 = 5.8 nM T86130 CQSH61 44461614 IC50 = 1600 nM T86130 CT16XO 44461624 IC50 = 100 nM T86130 CEBV54 44461633 IC50 = 11 nM T86130 CNZB87 44461659 IC50 = 450 nM T86130 C3XY2N 44461691 IC50 = 1.2 nM T86130 C3KZO9 44461700 IC50 = 49 nM T86130 CV6H2E 44461702 IC50 = 85 nM T86130 C75DRE 44461738 IC50 = 15 nM T86130 C46JYK 44461742 IC50 = 25 nM T86130 CJ3O2R 44461772 IC50 = 1.9 nM T86130 C37ZIL 44461783 IC50 = 6800 nM T86130 CR6K0X 44461787 IC50 = 0.3 nM T86130 C6NR7U 44461791 IC50 = 69 nM T86130 CECY94 44461792 IC50 = 890 nM T86130 C9BW3R 44461798 IC50 = 0.44 nM T86130 COTN73 44461809 IC50 = 0.42 nM T86130 CG63XE 44461810 IC50 = 16 nM T86130 C9KP0W 44461818 IC50 = 1.9 nM T86130 C85ALC 44461821 IC50 = 17 nM T86130 CUV91R 44461822 IC50 = 1.2 nM T86130 CPA74Y 44461824 IC50 = 1300 nM T86130 C9J2NM 44461832 IC50 = 3.3 nM T86130 CO3M5P 44461836 IC50 = 460 nM T86130 C81WRV 44461848 IC50 = 1.1 nM T86130 C8JCQ5 44561047 IC50 = 10 nM T86130 CDEJ98 44561562 IC50 = 10 nM T86130 CVB0M7 44561563 IC50 = 1616 nM T86130 CW6L8K 44580924 IC50 = 30 nM T86130 C7SUH8 44580925 IC50 = 378.5 nM T86130 CL04ER 44580926 IC50 = 490 nM T86130 CTZ7J4 44580927 IC50 = 4.41 nM T86130 CD2E9S 44580928 IC50 = 1.8 nM T86130 C60JSN 44580929 IC50 = 1070 nM T86130 CPVG97 44580930 IC50 = 1150 nM T86130 CTO41E 44580931 IC50 = 346.5 nM T86130 CT76BM 44604820 IC50 = 70 nM T86130 CY0R7W 44604821 IC50 = 4.4 nM T86130 C6J9TX 44604822 IC50 = 47 nM T86130 C4V5FN 44605030 IC50 = 1680 nM T86130 CCMR67 44605031 IC50 = 2.8 nM T86130 CRP3J6 44605032 IC50 = 138 nM T86130 C65LAB 44605033 IC50 = 12 nM T86130 CS3X8P 44605034 IC50 = 7.3 nM T86130 CY9F1E 44605241 IC50 = 20 nM T86130 C9UXR1 44605242 IC50 = 40 nM T86130 CD3XA9 44605243 IC50 = 1.9 nM T86130 C06DWR 44605244 IC50 = 2.7 nM T86130 CQ6GJ0 44605245 IC50 = 0.53 nM T86130 CBT94Y 44605422 IC50 = 8.5 nM T86130 C7U6MQ 44605423 IC50 = 2.6 nM T86130 CON35U 44605424 IC50 = 5 nM T86130 CV4DL2 44605425 IC50 = 204 nM T86130 C56FYN 44605619 IC50 = 2.7 nM T86130 CCT72M 44605620 IC50 = 7.5 nM T86130 CH75LV 44605621 IC50 = 128 nM T86130 C3N1FS 44605622 IC50 = 14 nM T86130 CQ2C8W 44605798 IC50 = 32 nM T86130 C64VMH 44605799 IC50 = 12 nM T86130 C2YA9X 44605800 IC50 = 6.4 nM T86130 C6SDP1 44605801 IC50 = 70 nM T86130 COGS45 44605971 IC50 = 2.9 nM T86130 CM58OC 44605972 IC50 = 241 nM T86130 CFR25V 45485799 IC50 = 3.1 nM T86130 CT8PH7 45485800 IC50 = 0.15 nM T86130 CI1OM4 45485801 IC50 = 0.27 nM T86130 C3C7DW 45485802 IC50 = 0.9 nM T86130 CHP37W 45485803 IC50 = 0.22 nM T86130 C08OHX 45485804 IC50 = 0.12 nM T86130 C9GOX0 45485805 IC50 = 0.24 nM T86130 CU0ZN8 45485806 IC50 = 0.1 nM T86130 CLFJ36 45485807 IC50 = 0.11 nM T86130 CZIA91 45485808 IC50 = 0.21 nM T86130 CI21LD 45485809 IC50 = 0.35 nM T86130 C8JRK2 45485810 IC50 = 0.22 nM T86130 CLA4C0 51346866 IC50 < 1 nM T86130 C3FK9V 52944365 IC50 = 0.022 nM T86130 CR0VI1 53317098 IC50 = 20 nM T86130 C2XIR7 53317680 IC50 = 8 nM T86130 C5YO8Q 53317712 IC50 = 32 nM T86130 CI5M9T 53318392 IC50 = 77 nM T86130 C7QWK8 53318393 IC50 = 75 nM T86130 CA3N7U 53319721 IC50 = 190 nM T86130 CTU86V 53319836 IC50 = 85 nM T86130 CMSZ29 53321012 IC50 = 130 nM T86130 CO4ES1 53322356 IC50 = 5 nM T86130 CO7Y9N 53326283 IC50 < 1 nM T86130 CD8KJ6 54686083 IC50 = 480 nM T86130 C9TZL8 56670195 IC50 = 2 nM T86130 C2L7DX 56671702 IC50 > 100000 nM T86130 C9VZ5T 56673720 IC50 = 4.5 nM T86130 C37IYH 56673727 IC50 = 1.27 nM T86130 C1D3YU 56677024 IC50 = 4100 nM T86130 C4H5QC 56677025 IC50 = 6 nM T86130 CWUD30 56677031 IC50 = 0.07 nM T86130 CDU79K 56678432 IC50 > 100000 nM T86130 C8UQ4J 56681774 IC50 = 20000 nM T86130 CGN1O4 56683691 IC50 = 105 nM T86130 C38ZTK 56835098 IC50 = 14100 nM T86130 CLY3O0 57391339 IC50 = 2.3 nM T86130 CF7V6D 57391340 IC50 = 487 nM T86130 C6RHB7 57391341 IC50 = 9.2 nM T86130 CHYV65 57391342 IC50 = 9 nM T86130 C07YKP 57391343 IC50 = 4 nM T86130 C1C6FM 57392592 IC50 = 36300 nM T86130 C36JEL 57393113 IC50 = 7.3 nM T86130 C9UWQ2 57393114 IC50 = 43 nM T86130 CT3AL8 57393115 IC50 = 59 nM T86130 CJH1C0 57394181 IC50 > 1000000 nM T86130 C0DJ9B 57394741 IC50 = 7 nM T86130 CQW75O 57394842 IC50 = 22 nM T86130 COJS48 57394843 IC50 = 432 nM T86130 CY0W4B 57394844 IC50 = 2.5 nM T86130 CCP9M4 57396072 IC50 = 2600 nM T86130 C4WH6P 57396074 IC50 = 169800 nM T86130 C3TWF2 57396501 IC50 = 2.6 nM T86130 CN7HX3 57396613 IC50 = 30 nM T86130 C1C2ZX 57396614 IC50 = 65 nM T86130 CR7C2I 57397874 IC50 = 123000 nM T86130 C2HN8S 57400043 IC50 = 900 nM T86130 C2LFD8 57401287 IC50 = 68400 nM T86130 C3ZH1K 57401732 IC50 = 3.6 nM T86130 CS2IB8 57401849 IC50 = 200 nM T86130 CK3WJ4 57402940 IC50 = 151400 nM T86130 C2ZD1U 57402941 IC50 = 97700 nM T86130 C80JUE 57403561 IC50 = 4.7 nM T86130 CYU4K8 58778354 IC50 = 1.1 nM T86130 CJF32X 58778988 IC50 = 3.7 nM T86130 CA82IB 69232792 IC50 = 140 nM T86130 C9QZG0 69335939 IC50 = 196 nM T86130 CSC75B 69335964 IC50 = 35 nM T86130 CSOG60 69336100 IC50 = 63 nM T86130 C6I8MK 69336784 IC50 = 87 nM T86130 CZEN52 69336954 IC50 = 123 nM T86130 C2SDK6 69337248 IC50 = 8 nM T86130 CO2M1D 69337579 IC50 = 18 nM T86130 CWU2B4 69667831 IC50 = 3500 nM T86130 C3T7XI 69667839 IC50 = 690 nM T86130 C30YPT 69667846 IC50 = 2900 nM T86130 C81THR 69667878 IC50 = 980 nM T86130 C0ADC9 69667917 IC50 = 370 nM T86130 C1PY8S 69667924 IC50 = 2700 nM T86130 CP6KM0 69667981 IC50 = 4 nM T86130 CW8HC3 69668030 IC50 = 1200 nM T86130 CPV02R 69668050 IC50 = 830 nM T86130 CCI6G2 69668079 IC50 = 4800 nM T86130 C97YHD 69668157 IC50 = 1200 nM T86130 CNI1B6 69668200 IC50 = 890 nM T86130 CQU6S8 69668225 IC50 = 160 nM T86130 C7JUG1 69668301 IC50 = 1200 nM T86130 C8XE9I 69668515 IC50 = 430 nM T86130 CNTU56 69668541 IC50 = 2700 nM T86130 C3M2HW 69668634 IC50 = 760 nM T86130 CO7KD2 69668636 IC50 = 1800 nM T86130 CS14BF 69668659 IC50 = 290 nM T86130 CMZ3H5 69668691 IC50 = 1500 nM T86130 CK4D7V 69668797 IC50 = 1900 nM T86130 C28KZD 69714759 IC50 = 225 nM T86130 CFU54E 69714767 IC50 = 48 nM T86130 CK5C3Q 69715313 IC50 = 269 nM T86130 CP5Y8I 69715941 IC50 = 267 nM T86130 C0G7XN 69716544 IC50 = 366 nM T86130 CJY8G4 71508676 IC50 = 16 nM T86130 CHW29E 71508677 IC50 = 4.3 nM T86130 CP7F3I 71508705 IC50 = 1.8 nM T86130 CQ7G3F 71508706 IC50 = 1.7 nM T86130 C1WU4J 71508734 IC50 = 1.7 nM T86130 CQGJ73 71508735 IC50 = 1.7 nM T86130 C4KXG2 71508736 IC50 = 3.6 nM T86130 C43KZG 71508737 IC50 = 3.7 nM T86130 C6ZCM5 71508738 IC50 = 202 nM T86130 CT2OV8 71508774 IC50 = 5.5 nM T86130 C05QCD 71508775 IC50 = 6.8 nM T86130 CH80VD 71508776 IC50 = 1.7 nM T86130 CM3WZ8 71508777 IC50 = 2.2 nM T86130 CTPE64 71508813 IC50 = 9 nM T86130 CS3L5W 71508814 IC50 = 4.2 nM T86130 C76YRK 71552171 IC50 = 820 nM T86130 C60QOE 71552172 IC50 = 112 nM T86130 C6YE4B 71552173 IC50 = 463 nM T86130 CJS16Z 71553006 IC50 = 25 nM T86130 C93EGS 71553082 IC50 = 64 nM T86130 C4OT8U 71553149 IC50 = 215 nM T86130 CC43TU 71562480 IC50 = 1400 nM T86130 C6YS7E 71716980 IC50 = 560 nM T86130 CA8FW2 71716981 IC50 = 255 nM T86130 C4HY2C 71717599 IC50 = 1450 nM T86130 CY13HN 71720011 IC50 = 246 nM T86130 CS0D7R 71727849 IC50 = 50.7 nM T86130 C6QJA2 71727850 IC50 = 97.1 nM T86130 CD1NH6 71727851 IC50 = 589.2 nM T86130 C1B7MR 71727976 IC50 = 366.4 nM T86130 CEG34M 71727977 IC50 = 17224.7 nM T86130 CU5CB6 71727978 IC50 = 80 nM T86130 CW6T4H 71728104 IC50 = 9.5 nM T86130 CMC5Q3 71728105 IC50 = 23388.7 nM T86130 CN3QT4 71728106 IC50 = 158.2 nM T86130 CQ8HY9 71728107 IC50 = 128.2 nM T86130 C59QKD 71728220 IC50 = 10.3 nM T86130 CB95ZS 71728221 IC50 = 37.9 nM T86130 C9R1BP 71728222 IC50 = 887.6 nM T86130 CW5GD8 73347006 IC50 = 40 nM T86130 CS9TD3 73347541 IC50 = 23.3 nM T86130 CNB39H 73356133 IC50 = 5 nM T86130 CQO2M7 76310621 Ki > 100000 nM T86130 CD46SJ 76321533 IC50 = 93 nM T86130 CS3Q1U 76332374 Ki > 100000 nM T86130 CNF56Z 76332375 Ki = 60 nM T86130 CEQ2Z4 76336006 Ki = 2400 nM T86130 CQH1Z7 90667312 IC50 = 703000 nM T86130 C7RLE0 90667313 IC50 = 208900 nM T86130 C7Q9GI 90667314 IC50 = 138000 nM T86130 CN9JF1 90667315 IC50 = 102300 nM T86130 C5HL9F 90667316 IC50 = 33100 nM T86130 CM5NK9 90667317 IC50 = 24300 nM T86130 CI35NK 90667318 IC50 = 151400 nM T86130 CVAY26 90667319 IC50 = 81300 nM T86130 C49WQN 90667320 IC50 = 97700 nM T86130 CS3T2Z 90667321 IC50 = 105900 nM T86130 CX3W0N 90667322 IC50 = 24500 nM T86130 CUL79M 90667323 IC50 = 38900 nM T86130 C46YXH 90667324 IC50 > 500000 nM T86130 C6YPL0 90667325 IC50 = 146200 nM T86130 CNH0W3 90667326 IC50 = 64600 nM T86130 CFT4Q1 90667327 IC50 = 81300 nM T86130 C73XBN 90667328 IC50 = 79400 nM T86130 C25QRP 90667329 IC50 = 190100 nM T86130 CKRV51 122181677 IC50 = 110 nM T86130 C2Q6TI 122181678 IC50 = 250 nM T86130 C0CNR5 122181679 IC50 > 1000 nM T86130 CV7DK0 122181680 IC50 = 10 nM T86130 C0O2HZ 122181681 IC50 > 1000 nM T86130 CWY3V2 122181682 IC50 = 62 nM T86130 C21ACR 133633869 EC50 = 255 nM T86130 C9T0FH 135416233 IC50 = 12 nM T86130 CPU86F 135438774 IC50 > 20000 nM T86130 C3JVT0 136152923 IC50 > 20000 nM T86130 C75GFR 154734316 IC50 = 1.39 nM T86130 CRI0W1 154734317 EC50 = 12.9 nM T86130 C8ZUJ5 154734319 IC50 > 1000 nM T86130 CAM96T 155519972 EC50 = 976 nM T86130 C6TCP5 155546837 IC50 > 1000 nM T86130 CY8S2L 155569251 IC50 > 1000 nM T86130 CZ9D2V 90645090 IC50 >= 100000 nM T86130 CWA6N4 90645092 IC50 >= 100000 nM T86130 D06LKH 123811 IC50 > 1000000 nM T86130 D08XWS 11226207 IC50 = 4.4 nM T86130 D09XED 11433918 IC50 = 0.15 nM T86130 D0A0JM 10120218 EC50 = 5.4 nM T60693 D00KHM 16362 IC50 = 990 nM T60693 D00UYE 4058 IC50 = 2370 nM T60693 D01KQA 5311304 Ki = 2.2 nM T60693 D02NSF 5284604 Ki = 25.3 nM T60693 D02RXG 6918287 EC50 = 0.0082 nM T60693 D03DIG 5284371 IC50 = 15000 nM T60693 D03SKD 5284603 EC50 = 16000 nM T60693 D04JEE 4946 EC50 > 5011.87 nM T60693 D04JHN 5284570 Ki = 2.8 nM T60693 D05GKD 33741 Ki > 10000 nM T60693 D05VIL 5284594 Ki = 0.083 nM T60693 D06AWE 644073 Ki = 0.04 nM T60693 D09OJQ 4095 IC50 = 512 nM T60693 D0CQ0Z 33630 Ki = 1000 nM T60693 D0D7KC 5488548 Ki = 100 nM T60693 D0E1WI 3345 Ki = 196.5 nM T60693 D0PG8O 5360515 Ki = 0.042 nM T60693 D0T3HY 5359272 Ki = 2.3 nM T60693 D0WE3O 5288826 Ki = 6.9 nM T60693 D0X3FX 5284596 Ki = 0.25 nM T60693 D0X5KF 5284569 Ki = 260 nM T60693 D0X9RG 5361092 Ki = 0.12 nM T60693 D00HBR 5486554 Ki = 0.48 nM T60693 D03PJU 62156 Ki = 43.1 nM T60693 D06ENM 66553195 EC50 = 1400 nM T60693 D06EXA 128563 EC50 = 0.015 nM T60693 D07TQN 179340 EC50 = 0.5 nM T60693 D07YHM 44129648 Ki = 0.597 nM T60693 D09ALE 60768 Ki = 0.27 nM T60693 D0G4YZ 11653141 Ki = 2200 nM T60693 D0LI1C 44469321 IC50 > 10000 nM T60693 D0N1HW 5311200 Ki > 10000 nM T60693 D0T0ZW 11667832 Ki = 0.23 nM T60693 D0V5WL 443363 Ki > 10000 nM T60693 D0W4YO 16131448 EC50 = 78.5 nM T60693 D0C2QF 9906198 Ki = 0.32 nM T60693 D0M1YN 5311194 Ki > 400 nM T60693 D0N1RG 9805452 Ki = 20 nM T60693 D0X6SZ 9826034 Ki = 0.15 nM T60693 D00ACC 9844019 Ki > 400 nM T60693 D06DZI 107780 Ki > 10000 nM T60693 D0A1KU 11683187 Ki = 3000 nM T60693 D0K5KL 119029 IC50 = 20 nM T60693 D0LX5D 5487663 Ki = 270 nM T60693 D0M7BW 3505 IC50 = 0.018 nM T60693 C21VAX 1223 Ki = 0.04 nM T60693 CAG0J1 5523 Ki = 14 nM T60693 C5H9CN 9287 Ki > 10000 nM T60693 CZC17M 9669 Ki = 2.2 nM T60693 CR6K8X 20906 IC50 = 157 nM T60693 CNZD18 36381 Ki = 488 nM T60693 C6E8DS 62513 Ki > 10000 nM T60693 CBGO28 70419 Ki = 196 nM T60693 CX5R6B 71420 IC50 = 155 nM T60693 CYKE31 104920 IC50 = 2140 nM T60693 C9NJK8 114876 Ki = 8.13 nM T60693 CQYC47 121999 Ki = 404 nM T60693 CDM08R 124716 Ki = 63 nM T60693 C7USG2 132913 Ki = 833 nM T60693 CB8Y9H 134131 Ki = 17 nM T60693 CVL3Z7 190901 Ki = 5.8 nM T60693 C4LEU1 191408 Ki > 10000 nM T60693 CX2I7G 356604 Ki = 15 nM T60693 C3HB4V 416359 IC50 = 110 nM T60693 CBLC72 457967 EC50 = 110 nM T60693 CR45EB 644177 Ki = 1.8 nM T60693 C3VFW0 715222 IC50 = 2650 nM T60693 CZN6S9 743974 EC50 > 100000 nM T60693 C6BDH3 780684 EC50 = 39 nM T60693 C6B0TP 1121183 EC50 = 7 nM T60693 CF4U0B 2162753 EC50 = 2000 nM T60693 C16UJC 2571306 Ki = 912.01 nM T60693 CAO06Q 2796048 IC50 = 376 nM T60693 C5M4BI 2846514 Ki = 6600 nM T60693 CLXC53 3000341 Ki = 1910 nM T60693 CAQ2J0 3034396 Ki = 198 nM T60693 C2TAD3 3036289 Ki = 0.2 nM T60693 CLB7W5 3037886 Ki = 9.9 nM T60693 CH0Z2R 3037926 Ki = 0.07 nM T60693 C5HDK8 3041260 Ki = 57.4 nM T60693 C5K7GJ 3054741 EC50 = 3.3 nM T60693 C8OHF0 3081578 Ki = 2.5 nM T60693 CMKU43 3086068 Ki = 4.96 nM T60693 C19ESC 3086114 IC50 = 13.09 nM T60693 CDIN98 3132840 EC50 = 3400 nM T60693 CJ6D8N 3342390 IC50 = 138 nM T60693 CQ6MW0 3655995 Ki = 84.5 nM T60693 C0YXV3 3676358 Ki > 10000 nM T60693 CY7LK9 4491166 Ki = 0.62 nM T60693 CANE93 4545429 Ki = 0.04 nM T60693 CO3U4Y 4736697 Ki = 83.18 nM T60693 CKLG29 5244802 IC50 = 11 nM T60693 C2O3TW 5282407 IC50 = 9480 nM T60693 CJX28Y 5311003 Ki = 2.4 nM T60693 CLW4B1 5311340 Ki = 1057 nM T60693 CRM46F 5320227 Ki > 10000 nM T60693 C2HPQ4 5462505 Ki = 22.8 nM T60693 C17RBP 5486940 Ki = 15.1 nM T60693 CJ7IE6 5487695 Ki = 128 nM T60693 CCMZ86 5491688 Ki > 3000 nM T60693 CZ4TM3 5492619 Ki = 5430 nM T60693 CI7L4R 5492830 Ki = 3090 nM T60693 C9LJ2K 5493351 Ki = 0.648 nM T60693 CJ5Z0D 6324613 Ki = 0.39 nM T60693 CB3M8S 6331636 Ki = 31.7 nM T60693 C5AL8S 6445230 EC50 = 0.025 nM T60693 CQML02 6603856 IC50 = 0.02 nM T60693 CED0X6 6604724 EC50 = 46 nM T60693 CM6VF8 6734379 IC50 = 2235 nM T60693 CFTO93 6918704 Ki = 16 nM T60693 CD49UV 9797246 Ki = 252 nM T60693 CNO0W4 9799433 Ki = 82.4 nM T60693 C8ANR0 9801260 IC50 = 7017 nM T60693 C5RNW7 9801830 IC50 = 2.3 nM T60693 C3V7JB 9802297 Ki = 124 nM T60693 CPG57N 9803475 Ki > 400 nM T60693 CX7DO4 9806799 Ki = 871 nM T60693 CP5IE7 9821780 Ki = 0.058 nM T60693 CJ72XV 9822639 Ki = 24 nM T60693 CXV1R9 9822756 IC50 = 1.5 nM T60693 CE6NF9 9823363 IC50 = 1400 nM T60693 C70KEP 9824565 Ki = 747 nM T60693 CR54GJ 9824976 Ki = 163 nM T60693 CBXY90 9828569 IC50 = 0.11 nM T60693 CW1T4D 9839245 Ki = 0.06 nM T60693 C4QFZ6 9841259 IC50 = 7470 nM T60693 CKVQ31 9843334 Ki = 171 nM T60693 C6Y7NA 9844540 Ki = 635 nM T60693 CH06GL 9848989 IC50 = 1.2 nM T60693 CKD2H4 9848990 Ki = 0.067 nM T60693 CBMN05 9865332 Ki = 66 nM T60693 CLQ6Z8 9866158 Ki = 116 nM T60693 CL26PE 9866175 Ki > 890 nM T60693 CQ4LC2 9872676 Ki = 1960 nM T60693 CPYK08 9887195 IC50 = 2600 nM T60693 CVH87F 9887566 Ki = 1448 nM T60693 CJF8C2 9890982 IC50 = 4.8 nM T60693 CGQA14 9891527 IC50 = 0.2 nM T60693 C5BC4P 9902874 Ki = 6212 nM T60693 CUN81Q 9905249 Ki > 10000 nM T60693 CX3CM8 9905428 Ki = 42.7 nM T60693 CB6C8L 9911987 Ki = 744 nM T60693 CJFO67 9912633 EC50 = 1.1 nM T60693 CZT2J0 9927928 Ki = 37.92 nM T60693 C26DMO 9928857 Ki = 36.5 nM T60693 C3PGN9 9931141 EC50 = 0.4 nM T60693 CQU6D0 9931316 IC50 = 0.47 nM T60693 CVK0R1 9932084 IC50 = 0.9 nM T60693 CM3B5E 9932532 Ki > 890 nM T60693 C2U8XH 9932834 Ki = 109 nM T60693 CYZW21 9932852 EC50 > 30 nM T60693 C9MK3B 9934232 Ki = 5887 nM T60693 CUBQ95 9937777 Ki = 254 nM T60693 CO7BI9 9940052 Ki = 0.18 nM T60693 C4FD7V 9947044 Ki = 10.7 nM T60693 CG9ER5 9947155 Ki > 2000 nM T60693 C5S3RH 9949205 Ki = 11.92 nM T60693 COFT18 9951673 Ki = 1136 nM T60693 C3GXH0 9954388 Ki = 44.2 nM T60693 CT8C2X 9958643 Ki = 278 nM T60693 CE3CJ4 9969865 Ki > 2000 nM T60693 CJG3Q1 9974346 Ki = 0.93 nM T60693 C1B2JR 9976188 Ki > 500 nM T60693 C71QEP 9981894 Ki = 3.7 nM T60693 C0H3JC 9984459 Ki = 25 nM T60693 C2GI1Q 9984781 Ki = 0.3 nM T60693 C2WJL0 9990996 Ki = 345 nM T60693 CDPW27 9997232 Ki = 0.93 nM T60693 CAGL19 9997843 Ki = 5.3 nM T60693 CN2F1U 10001960 IC50 = 5350 nM T60693 CL9QS0 10004950 IC50 = 2.1 nM T60693 C9CP0Q 10005080 EC50 = 0.1 nM T60693 CQ43EZ 10016044 Ki = 0.07 nM T60693 CV7R9F 10020040 Ki > 10000 nM T60693 C4N8YE 10020165 Ki = 229 nM T60693 CL38DM 10021831 Ki = 122.2 nM T60693 C25DYT 10022859 Ki = 25.12 nM T60693 C0O9EM 10024658 IC50 = 8.7 nM T60693 C1PGE2 10031234 Ki > 1000 nM T60693 C61SQU 10033525 IC50 = 6.29 nM T60693 CFOK60 10042904 Ki = 148 nM T60693 CE0VX6 10044490 Ki = 0.41 nM T60693 C4CXP1 10053267 EC50 = 0.12 nM T60693 C8WE1N 10055958 IC50 = 7330 nM T60693 C1ED3S 10070066 IC50 = 2.7 nM T60693 CS3UK5 10074239 Ki = 94.2 nM T60693 CO8P3K 10076169 EC50 = 0.34 nM T60693 CQVA98 10078468 Ki = 0.076 nM T60693 CW3GI2 10090773 Ki = 0.58 nM T60693 CNAB97 10095688 EC50 = 3000 nM T60693 C7YCF1 10109899 Ki = 519 nM T60693 CJNE19 10110916 Ki > 2000 nM T60693 C76MVA 10111186 Ki > 2000 nM T60693 CWEC34 10114637 Ki > 2000 nM T60693 C45XQC 10117927 Ki = 0.44 nM T60693 C40BMF 10133108 Ki = 1394 nM T60693 CP1SO7 10134077 Ki > 10000 nM T60693 CEG0M4 10134217 Ki > 2000 nM T60693 C3ZTU0 10137134 Ki = 1672 nM T60693 C83KDV 10137876 Ki > 2000 nM T60693 C8E9KP 10139672 Ki > 2000 nM T60693 CI3PJ6 10149623 Ki > 10000 nM T60693 CQGE97 10150001 Ki = 660 nM T60693 CF85VW 10150089 Ki > 10000 nM T60693 C76SOW 10150260 Ki = 1232 nM T60693 CTO0N5 10158555 Ki = 150 nM T60693 CWM2X6 10160920 Ki > 2000 nM T60693 C67SZC 10171702 Ki > 10000 nM T60693 CDV15J 10172398 Ki = 150 nM T60693 CJN21A 10178311 Ki > 10000 nM T60693 CK5HG3 10179322 Ki > 4652 nM T60693 CHC6K9 10179323 Ki = 201 nM T60693 C5RO6K 10182346 Ki > 2000 nM T60693 C2SP7U 10183838 Ki = 346 nM T60693 CB0TE3 10186312 Ki = 0.36 nM T60693 CNZL85 10193971 Ki = 6488 nM T60693 CN79QX 10194236 Ki = 1634 nM T60693 CWC8L1 10199945 IC50 = 160 nM T60693 C12NGT 10199984 Ki > 2000 nM T60693 C85DFV 10201299 Ki = 108 nM T60693 CV1T7R 10202241 Ki > 2000 nM T60693 C9ZCT0 10206319 Ki = 725 nM T60693 CJ74DP 10207990 Ki = 0.53 nM T60693 C02IUS 10214859 Ki = 1500 nM T60693 CYB0H9 10221539 IC50 = 60 nM T60693 CRGJ86 10224456 IC50 = 700 nM T60693 C2MQS5 10227615 Ki = 88 nM T60693 C6LQH4 10245350 Ki = 5.7 nM T60693 CO8TH6 10248394 Ki = 1.1 nM T60693 CF37AI 10249808 Ki = 0.064 nM T60693 CZ0C5T 10252647 Ki = 543 nM T60693 CR4C1F 10253032 Ki = 6 nM T60693 C4RX1A 10256503 EC50 = 0.17 nM T60693 CH31DX 10267394 Ki > 10000 nM T60693 C6YKB9 10273543 Ki = 2.8 nM T60693 C8PL7B 10274330 Ki > 2000 nM T60693 C89KBW 10286378 Ki > 10000 nM T60693 CDP01X 10286440 Ki = 13130 nM T60693 C1FE9H 10286996 Ki = 4015 nM T60693 CJ14VU 10291377 Ki = 1701 nM T60693 CKO2I1 10297473 Ki = 25 nM T60693 CF4VO2 10308746 Ki > 10000 nM T60693 CU89JD 10314060 Ki > 10000 nM T60693 CFHC64 10315026 Ki = 7.5 nM T60693 CQD21X 10315939 Ki = 68.5 nM T60693 CM12XP 10316899 Ki = 0.065 nM T60693 CX16OB 10319320 IC50 = 1.1 nM T60693 C68AST 10320450 Ki = 68 nM T60693 C1ENR2 10323169 Ki = 15 nM T60693 CA4KJ5 10323346 EC50 = 96.2 nM T60693 CUJ0N2 10331735 Ki = 66 nM T60693 CH14KO 10334091 EC50 = 9.7 nM T60693 C54WJL 10337395 Ki = 0.49 nM T60693 C0YB6G 10338942 IC50 = 22 nM T60693 CRY8O2 10340520 IC50 = 15 nM T60693 C63GNX 10342726 EC50 = 0.2 nM T60693 C3P0LR 10345440 EC50 = 0.26 nM T60693 CJXM25 10347927 EC50 = 0.54 nM T60693 CPJ5N4 10349271 Ki = 0.57 nM T60693 CPO17B 10351514 IC50 = 12.14 nM T60693 CM6N1T 10358054 Ki = 49 nM T60693 C0ZF8R 10366960 IC50 = 640 nM T60693 CFZ52M 10372345 Ki = 0.39 nM T60693 C7GK4U 10378392 Ki > 10000 nM T60693 CAYF18 10385808 Ki > 2000 nM T60693 CYD30U 10387038 Ki = 45.01 nM T60693 C95EWP 10395965 Ki = 105 nM T60693 CWK4O1 10406239 Ki = 2.3 nM T60693 CTA8Q0 10407144 Ki = 22.7 nM T60693 CX6ZH1 10408431 IC50 = 37 nM T60693 CN5TB6 10408752 Ki = 0.3 nM T60693 CI17TP 10410240 Ki = 0.13 nM T60693 CK2C6S 10410389 Ki = 220 nM T60693 CYWF17 10412617 IC50 > 10000 nM T60693 C5S0UF 10413389 Ki = 8.6 nM T60693 C6LBC5 10415925 Ki > 10000 nM T60693 C1U6NG 10430432 Ki = 0.58 nM T60693 CYHC38 10430819 Ki = 281.84 nM T60693 CY54PU 10431414 Ki = 3722 nM T60693 CON12X 10435156 Ki = 13.8 nM T60693 CQ4M0D 10443502 Ki = 184 nM T60693 C7AQ0G 10449693 Ki = 95 nM T60693 CZ6I9V 10451761 IC50 = 440 nM T60693 CV14CY 10452891 IC50 = 2290 nM T60693 C0M9AN 10461299 Ki = 0.32 nM T60693 CKMN08 10475466 Ki = 26 nM T60693 CE3HW8 10476369 IC50 = 1.4 nM T60693 CEF2O6 10478367 Ki > 10000 nM T60693 C29OZW 10484384 Ki = 23.6 nM T60693 CE2LD8 10486131 Ki = 4.6 nM T60693 CP72JI 10499145 IC50 > 10000 nM T60693 C1DI7F 10500922 Ki = 149 nM T60693 CGCP09 10501573 IC50 > 10000 nM T60693 C90DEM 10504545 Ki = 26.2 nM T60693 C0G2QX 10508302 Ki = 36.3 nM T60693 CJ2BC7 10525105 IC50 = 4906 nM T60693 CDGM01 10525171 IC50 > 10000 nM T60693 C8FB2A 10527816 Ki = 13.49 nM T60693 C41JWE 10546813 IC50 = 4530 nM T60693 CDK8W2 10548749 Ki = 16.4 nM T60693 CJ1TU0 10549849 IC50 = 980 nM T60693 CKP6E2 10550601 IC50 = 1330 nM T60693 C71YXH 10553426 Ki = 0.49 nM T60693 CKT1L0 10569964 IC50 > 10000 nM T60693 C8E1UH 10570940 IC50 > 10000 nM T60693 CLU72B 10572649 IC50 > 10000 nM T60693 C54EOA 10572810 Ki = 48 nM T60693 CD9JB5 10574643 Ki = 40.1 nM T60693 C28WNJ 10574908 Ki = 1.52 nM T60693 CQ74CO 10593778 Ki = 161 nM T60693 CT60BQ 10594839 IC50 > 8900 nM T60693 CY6D1C 10596575 IC50 > 10000 nM T60693 C2FL8C 10598391 IC50 > 10000 nM T60693 C2CF1X 10598392 IC50 > 10000 nM T60693 C71RMT 10599027 Ki = 0.5495 nM T60693 CHV5D1 10601891 Ki = 28.8 nM T60693 CS84IW 10618605 Ki = 46.3 nM T60693 CK96NW 10618862 IC50 > 10000 nM T60693 C62MNC 10620493 IC50 = 7574 nM T60693 CIM8S1 10620902 IC50 = 1660 nM T60693 CCV14H 10642101 IC50 = 724 nM T60693 C3CHZ0 10642670 IC50 > 10000 nM T60693 C4XYH5 10644815 IC50 = 3160 nM T60693 C8ZU7I 10644995 IC50 > 5600 nM T60693 CF36MK 10645976 Ki = 0.7 nM T60693 CPC52U 10646744 Ki = 16.4 nM T60693 C10KTE 10646745 Ki = 17.5 nM T60693 CFC5R6 10668838 IC50 = 6140 nM T60693 CA0M1N 10690216 IC50 = 6970 nM T60693 CGPT20 10692042 IC50 > 10000 nM T60693 CHC1I4 10697286 Ki = 52 nM T60693 C5U4ZP 10713071 IC50 > 10000 nM T60693 C2RN9F 10713623 Ki = 17 nM T60693 C8XB3K 10714523 Ki = 44 nM T60693 C2W9PN 10714960 IC50 = 8340 nM T60693 CUAC76 10718278 Ki = 49 nM T60693 C8D2PI 10718445 Ki = 1.31 nM T60693 CV8K3J 10720494 Ki = 340 nM T60693 CS82CN 10739828 IC50 > 10000 nM T60693 CAT04G 10741016 IC50 = 3160 nM T60693 C8RW7M 10742582 Ki = 27.8 nM T60693 CF61KY 10742765 Ki = 78.6 nM T60693 C4BJ9L 10760345 IC50 > 10000 nM T60693 CR4H2D 10760626 IC50 > 10000 nM T60693 C0PT3I 10762996 IC50 = 3967 nM T60693 CN05WO 10763594 Ki = 89 nM T60693 CIT9X3 10771171 Ki = 1367 nM T60693 CDJP34 10783436 IC50 = 12 nM T60693 CB0JQ9 10785784 IC50 = 2610 nM T60693 C54YIB 10786358 IC50 > 10000 nM T60693 CSXE56 10787424 IC50 = 4270 nM T60693 C2O0HR 10808721 IC50 > 10000 nM T60693 C9G7LT 10809678 IC50 > 10000 nM T60693 C3ZT7Y 10810430 Ki = 3160 nM T60693 CS3Y4G 10832076 IC50 = 32 nM T60693 CMVI50 10832445 Ki = 47.1 nM T60693 C9WI5X 10833535 IC50 > 10000 nM T60693 CPG23C 10836379 Ki = 47.3 nM T60693 C4IT2B 10837001 Ki = 17 nM T60693 CFP68N 10872951 IC50 = 9380 nM T60693 C7PR6B 10874095 IC50 = 1.3 nM T60693 CWL1K9 10874724 IC50 = 3580 nM T60693 CH4WY8 10883143 Ki = 0.25 nM T60693 C4ARK1 10883642 IC50 > 10000 nM T60693 C0H1TJ 10884365 IC50 = 1480 nM T60693 C9Y8OS 10884964 IC50 = 307 nM T60693 CB2QL0 10885771 IC50 = 7240 nM T60693 CR2D0K 10893581 IC50 = 521 nM T60693 CE6NR5 10893607 IC50 > 10000 nM T60693 C0LM2D 10893958 IC50 = 37 nM T60693 CF61NU 10895676 IC50 = 4030 nM T60693 CWJL70 10905740 IC50 = 32 nM T60693 CX65PW 10907460 IC50 = 4120 nM T60693 CQ62UO 10918307 IC50 = 333 nM T60693 CA86IC 10926896 Ki = 0.4467 nM T60693 CT79NZ 10927276 IC50 = 617 nM T60693 C4TSV6 10927662 Ki = 131.83 nM T60693 C1TSN4 10928037 Ki = 131.83 nM T60693 CR17TE 10928590 IC50 = 1060 nM T60693 CTN91R 10929002 IC50 = 1010 nM T60693 C9M2JE 10929207 IC50 = 6570 nM T60693 CT5UO7 10937810 Ki = 257.04 nM T60693 CU09AV 10937901 IC50 = 1.7 nM T60693 C6VBL1 10938869 Ki = 0.47 nM T60693 CM0OS2 10939174 IC50 = 2145 nM T60693 C6WQ3H 10939958 IC50 > 10000 nM T60693 CN7XS4 10948527 IC50 = 56.1 nM T60693 CSLT97 10949380 IC50 = 2.9 nM T60693 CCUE70 10950205 IC50 = 6540 nM T60693 C9FYG3 10950562 Ki = 512.86 nM T60693 C48NDC 10950714 IC50 > 10000 nM T60693 CKR58N 10951763 Ki = 16.2 nM T60693 CHK23I 10961428 Ki = 169.82 nM T60693 C1Y9ID 10971999 Ki = 0.31 nM T60693 C2HP7F 10981761 IC50 = 104 nM T60693 C32ZYJ 10982772 EC50 = 1.4 nM T60693 CMY56Q 10985930 Ki = 79.4 nM T60693 CSZ6R2 10985963 Ki = 6.61 nM T60693 C96ULE 10992239 IC50 = 2510 nM T60693 CD5V9L 10992895 IC50 = 996 nM T60693 C91NTI 11003763 IC50 = 1450 nM T60693 CJ6C9K 11003971 IC50 = 1740 nM T60693 C8Q6YE 11004121 Ki = 26.92 nM T60693 CJC9K4 11005810 IC50 = 1980 nM T60693 C3V7LT 11014751 Ki = 56.23 nM T60693 C8CP6J 11016127 IC50 = 2.8 nM T60693 C0VKL9 11016305 Ki = 0.153 nM T60693 C3WE6J 11024236 IC50 = 764 nM T60693 CC45BL 11025925 IC50 = 2280 nM T60693 CB7N1P 11035765 IC50 = 507 nM T60693 C0DE3C 11036499 Ki = 0.53 nM T60693 CUI3F2 11046929 IC50 = 270 nM T60693 C6EBF3 11048769 IC50 = 1810 nM T60693 C57NRV 11051174 Ki > 100000 nM T60693 CL8Z9G 11058283 Ki = 3190 nM T60693 CFJG64 11059058 IC50 = 284 nM T60693 CL9Y8H 11059305 IC50 = 797 nM T60693 C2ASJ3 11070421 Ki = 1.82 nM T60693 CG41BK 11071079 IC50 = 4230 nM T60693 C81MOC 11071091 IC50 = 2200 nM T60693 CWAB48 11071778 Ki = 6400 nM T60693 C5ZP8L 11082539 Ki > 10000 nM T60693 CS4BM0 11090195 IC50 = 1070 nM T60693 C49OUP 11090735 Ki = 4.34 nM T60693 CR0TL9 11091522 IC50 = 64.6 nM T60693 CA68BR 11091606 Ki = 0.3 nM T60693 CO08EV 11091686 IC50 = 5070 nM T60693 C6HIQ0 11092200 IC50 > 10000 nM T60693 C7WB6K 11094406 Ki = 10.7 nM T60693 CONE61 11104644 Ki = 5600 nM T60693 CF0SV1 11112699 IC50 = 321 nM T60693 C7DE0U 11113605 IC50 = 2820 nM T60693 C0RJ9M 11120930 Ki = 418 nM T60693 CJ25OQ 11122114 IC50 = 3550 nM T60693 C3CGB7 11123013 IC50 = 394 nM T60693 CDU0E5 11123873 Ki = 147.91 nM T60693 C6P5EL 11129476 Ki = 3470 nM T60693 C9WXY1 11132954 Ki > 10000 nM T60693 CN8UZ0 11136722 Ki = 60.3 nM T60693 C04HTO 11139094 IC50 > 10000 nM T60693 CIL4S3 11140284 Ki = 565 nM T60693 CU6PV0 11143820 IC50 = 5.7 nM T60693 CP96WD 11145858 EC50 = 11.5 nM T60693 CPW06I 11146107 Ki = 1600 nM T60693 C10FGZ 11149261 Ki = 232 nM T60693 C4NAJ5 11154544 Ki = 42 nM T60693 CE6N5V 11157443 Ki = 0.63 nM T60693 C67ZFK 11158498 Ki = 4.2 nM T60693 CJO8S0 11163232 Ki = 6.7 nM T60693 C26ENL 11164004 Ki = 202 nM T60693 C62WBJ 11165726 Ki = 74.4 nM T60693 C6A0JS 11166820 Ki = 284 nM T60693 C26PQJ 11167140 Ki = 1610 nM T60693 C49QZC 11179386 EC50 = 0.025 nM T60693 C16TCJ 11180190 Ki = 184 nM T60693 CPQ6A8 11180584 Ki = 2.38 nM T60693 CM9TV6 11181676 Ki = 1.2 nM T60693 CLE18Z 11184156 Ki = 263 nM T60693 CAKZ38 11184946 IC50 = 7400 nM T60693 CM6Q2S 11186913 Ki = 0.49 nM T60693 CF86JN 11188632 Ki = 3.8 nM T60693 CAZ30T 11188794 Ki = 2533 nM T60693 C90HXY 11190061 Ki = 468 nM T60693 CMRJ71 11191431 Ki = 93 nM T60693 CJL1R5 11198030 Ki = 207 nM T60693 CIG2Q9 11201660 Ki = 0.6 nM T60693 CGL3W7 11204993 Ki = 0.41 nM T60693 CKB01D 11212562 Ki = 890 nM T60693 CZ4US0 11215747 Ki = 2.41 nM T60693 CK8VG1 11220535 Ki = 82.3 nM T60693 C4QT5Y 11233481 Ki = 175 nM T60693 C7LD4V 11238343 Ki = 0.86 nM T60693 CA5T0Z 11238737 Ki = 0.66 nM T60693 C7DJ3L 11239327 Ki = 0.1 nM T60693 C8BO9A 11246669 Ki = 62 nM T60693 CMFI07 11248182 EC50 = 0.52 nM T60693 CWZP56 11256722 EC50 = 0.05 nM T60693 C5NCH0 11258701 Ki = 0.39 nM T60693 C1O5ZD 11262815 Ki = 0.59 nM T60693 CF4LV5 11264459 Ki = 333 nM T60693 CD19XU 11270347 Ki = 2.9 nM T60693 CMI48S 11271318 Ki = 2.3 nM T60693 C3G6PC 11273472 Ki = 1.61 nM T60693 C1B9ET 11274203 Ki = 0.7 nM T60693 CPBZ36 11274537 Ki > 5000 nM T60693 CA93LY 11280087 EC50 = 0.23 nM T60693 C5WYA8 11280721 Ki = 622 nM T60693 CG82EM 11280808 Ki = 1 nM T60693 CQ0FP3 11292970 Ki = 10 nM T60693 C5CK3W 11304200 Ki = 23 nM T60693 C59MLX 11305998 Ki = 120 nM T60693 CR4TD3 11307039 Ki = 24 nM T60693 CAWZ12 11308699 Ki = 3.4 nM T60693 CF60BC 11308721 Ki = 0.65 nM T60693 CAOJ05 11311787 Ki = 55.8 nM T60693 C8P5AT 11314197 Ki > 4000 nM T60693 C4FRH7 11315651 Ki > 400 nM T60693 CYT7N3 11316776 Ki > 1000 nM T60693 C9A1PL 11318909 Ki = 2.72 nM T60693 CR85OX 11319221 Ki = 6.96 nM T60693 CMK6Q8 11322246 Ki = 251 nM T60693 C5DBK1 11326750 IC50 > 10000 nM T60693 CJM7R5 11327115 Ki = 3869 nM T60693 C6BC9X 11327160 EC50 = 20.7 nM T60693 C9D4TI 11330655 Ki = 3.26 nM T60693 CI4SY0 11333521 Ki = 149 nM T60693 CIS8B5 11334123 Ki = 184 nM T60693 CIG49E 11339827 Ki = 65 nM T60693 C4C0OE 11341622 Ki = 64 nM T60693 CY0SV8 11349939 Ki = 343 nM T60693 CPSQ49 11350705 Ki = 0.11 nM T60693 C10YKF 11351067 Ki = 14 nM T60693 C48IOK 11351930 Ki = 26 nM T60693 CJ9P1G 11352435 Ki = 580 nM T60693 CXUI57 11353083 Ki = 38.7 nM T60693 C4CFD0 11358487 Ki = 1830 nM T60693 CB5F8T 11359173 Ki = 0.74 nM T60693 CLT47S 11364225 Ki = 0.07 nM T60693 C73GIN 11365113 Ki = 50 nM T60693 C6UZF7 11371415 Ki = 21.5 nM T60693 CGT16B 11372452 Ki = 0.27 nM T60693 CA19LC 11373068 Ki > 4652 nM T60693 C9HGE1 11374952 Ki = 430 nM T60693 CZS3E9 11376776 Ki = 1.42 nM T60693 C2E8MJ 11382472 Ki = 800 nM T60693 CX5Z0G 11383671 Ki = 0.53 nM T60693 CH50TV 11388486 Ki = 0.17 nM T60693 C5OIU1 11391288 Ki = 146 nM T60693 CR9V8F 11391721 Ki = 552 nM T60693 CT6Z0B 11393860 Ki = 55.1 nM T60693 CWA07Q 11397778 Ki = 6 nM T60693 C8XZ2G 11407876 Ki = 0.4 nM T60693 CN6G8I 11408550 Ki = 3.9 nM T60693 C0N5JW 11408724 Ki = 2.6 nM T60693 CBGR89 11419799 Ki = 19 nM T60693 C4S8GN 11421830 Ki = 2.74 nM T60693 CVBO48 11428892 Ki = 0.5 nM T60693 C3PSN6 11429436 Ki = 0.21 nM T60693 CS9G3B 11430490 Ki = 334 nM T60693 C3PD8Y 11430747 Ki = 5.7 nM T60693 CY5Z6D 11434336 Ki = 1.1 nM T60693 CKL6P9 11440457 Ki = 1.3 nM T60693 CSZ2F1 11440849 Ki = 505 nM T60693 C9R7AI 11444917 Ki = 3.91 nM T60693 C9KV1U 11451023 Ki = 52.1 nM T60693 CR4IV6 11453965 Ki = 16 nM T60693 C3M4ZJ 11455086 Ki = 250 nM T60693 C7UDE8 11461888 Ki = 31.7 nM T60693 CX4K6J 11463076 EC50 = 0.49 nM T60693 C7IXL1 11463580 Ki = 6 nM T60693 C24ZHJ 11463610 Ki = 280 nM T60693 CMU9K5 11464846 Ki > 400 nM T60693 CAO2E4 11465947 Ki = 96 nM T60693 CMV04H 11470285 Ki = 63.7 nM T60693 CO95HP 11474838 Ki = 830 nM T60693 C5GOD3 11477039 Ki = 1.5 nM T60693 C3T5SC 11479033 Ki = 4.8 nM T60693 C3BA5F 11480038 Ki = 4270 nM T60693 C4R8HV 11485758 Ki = 0.39 nM T60693 C4XU0O 11486901 Ki = 41 nM T60693 C1LJ5U 11487063 Ki = 1250 nM T60693 C5UR1M 11487946 Ki = 34 nM T60693 CA4PM8 11496383 EC50 = 6 nM T60693 CX6Q0I 11497325 Ki = 180 nM T60693 CYP08U 11509780 Ki = 55 nM T60693 C41MEV 11511090 IC50 = 950 nM T60693 C2E7LB 11511362 Ki = 200 nM T60693 C5LA3M 11521945 Ki = 350 nM T60693 CQ30PM 11525624 IC50 = 7900 nM T60693 C49XZQ 11526334 EC50 = 0.04 nM T60693 CB1K8W 11533999 Ki = 50 nM T60693 CF86WQ 11537712 Ki > 10000 nM T60693 CB2U5X 11540292 EC50 = 6 nM T60693 C8TZ9G 11544654 IC50 = 930 nM T60693 COF4K0 11544824 Ki > 10000 nM T60693 C64PNH 11546512 EC50 = 6.5 nM T60693 CHI36N 11547640 Ki = 70 nM T60693 CHI47M 11555262 Ki = 290 nM T60693 C2ZNA4 11558993 Ki > 10000 nM T60693 C97WYH 11559278 Ki = 57 nM T60693 CVI52T 11561040 Ki = 30 nM T60693 C0H8CM 11561655 Ki = 1.2 nM T60693 CO02FI 11562377 EC50 = 6 nM T60693 C3E4LV 11562400 Ki = 260 nM T60693 CWR06X 11581573 Ki = 51.6 nM T60693 CVA8L6 11583016 IC50 = 9600 nM T60693 CIJQ92 11583295 Ki = 42.3 nM T60693 C3PX0F 11584092 Ki = 440 nM T60693 CO0N2L 11591805 Ki = 0.85 nM T60693 CZA48L 11591838 Ki = 60 nM T60693 C9GPQ8 11595485 Ki > 10000 nM T60693 C1WBQ5 11597677 IC50 = 2300 nM T60693 CE4ZV5 11602862 Ki > 10000 nM T60693 C8RKH0 11619553 IC50 = 3700 nM T60693 CSYE45 11619680 EC50 = 6 nM T60693 CM8NO4 11628123 Ki = 90 nM T60693 C4ZD1X 11633324 IC50 = 6900 nM T60693 C2USB1 11655841 Ki = 15 nM T60693 CC1EZ6 11657075 Ki = 70 nM T60693 CQML27 11660069 Ki > 10000 nM T60693 CS91JQ 11666402 Ki > 10000 nM T60693 CXO5K2 11667199 Ki > 10000 nM T60693 C9XD2T 11677662 Ki = 0.29 nM T60693 CL05UW 11697184 Ki = 167 nM T60693 CW7QD2 11698381 EC50 = 6 nM T60693 C19DJE 11698420 EC50 = 6 nM T60693 C79XSW 11705263 Ki = 4 nM T60693 C4ULQ7 11710187 IC50 = 250 nM T60693 C4PXV7 11712760 EC50 = 6 nM T60693 CUG57V 11713930 Ki = 90 nM T60693 C8A2CG 11714559 Ki = 2.5 nM T60693 CC4SF3 11717551 Ki > 10000 nM T60693 COL07J 11728653 IC50 = 793 nM T60693 C7FSD3 11729952 IC50 = 1.5 nM T60693 C7PVL8 11730467 IC50 = 2150 nM T60693 CV3OY7 11733074 IC50 > 10000 nM T60693 CCN8E9 11742939 IC50 > 7600 nM T60693 CPG15O 11743399 IC50 > 1000 nM T60693 CG6SM0 11749794 Ki = 15 nM T60693 CBH0Y7 11753736 Ki = 0.95 nM T60693 CIDS04 11753832 EC50 = 9.6 nM T60693 CFRY36 11757207 Ki = 122 nM T60693 C3F5DX 11761059 IC50 = 311 nM T60693 CED7I5 11761926 Ki = 251.19 nM T60693 CEI7T9 11771732 Ki = 0.48 nM T60693 CC61WX 11773726 Ki = 1.27 nM T60693 CX27WK 11779453 EC50 = 2.8 nM T60693 C87CPT 11784022 Ki = 0.28 nM T60693 CJ7L9W 11784235 IC50 = 345 nM T60693 C1K0JF 11786990 Ki = 2.14 nM T60693 C7TLS3 11793476 IC50 > 10000 nM T60693 CJD95Z 11794240 IC50 > 10000 nM T60693 C1LJM6 11794241 IC50 > 10000 nM T60693 CG9HW8 11795019 Ki = 20.7 nM T60693 C5C8NP 11795327 Ki = 0.36 nM T60693 C60RKP 11796211 IC50 = 3870 nM T60693 C80ZJV 11797669 Ki = 35.1 nM T60693 C4SCZ1 11797670 Ki = 108 nM T60693 COSJ52 11811375 IC50 = 3100 nM T60693 CN9M8E 11811722 IC50 = 101 nM T60693 CXM98K 11811844 Ki = 3.77 nM T60693 CXY38K 11812228 IC50 = 1320 nM T60693 C8UE5W 11826819 Ki = 154.88 nM T60693 CC65TG 11827053 IC50 = 51.4 nM T60693 CS7W2V 11848793 Ki = 268 nM T60693 C65TDJ 11849246 IC50 = 39.1 nM T60693 CHV25L 11849247 EC50 = 1.8 nM T60693 CQ6P3Y 11849249 Ki = 2.4 nM T60693 CIKN38 11849282 Ki = 1.5 nM T60693 CR47EN 11849283 Ki = 9.9 nM T60693 C7SI8L 11849284 Ki = 2.3 nM T60693 CP8QH4 11849285 EC50 = 0.2 nM T60693 C7D2TB 11849360 Ki = 6.4 nM T60693 CK2RQ0 11849361 Ki = 2.5 nM T60693 CD39RT 11849364 EC50 = 9 nM T60693 C63YAV 11849365 IC50 = 12.1 nM T60693 CXLW54 11948707 Ki > 10000 nM T60693 CS0MC4 11950654 EC50 > 5000 nM T60693 CEVH83 12041054 Ki = 4.79 nM T60693 CJP1W3 12041055 Ki = 2.76 nM T60693 C5RD1S 12041056 Ki = 1.29 nM T60693 CQ1B6S 12048050 Ki = 620 nM T60693 CW40NY 12066967 Ki = 1980 nM T60693 CPA8N5 12066969 Ki = 190 nM T60693 CYCF29 12103026 IC50 > 10000 nM T60693 CT9KA1 12114808 Ki > 40000 nM T60693 CBK43E 12114809 Ki = 1080 nM T60693 C6IT0O 12191611 Ki > 10000 nM T60693 CYBD81 12191612 Ki = 14 nM T60693 CS5IZ8 12371110 Ki = 113 nM T60693 CSY9N8 12371111 Ki = 3776 nM T60693 CAR89Y 12994686 EC50 = 20 nM T60693 C4UB2W 13177879 Ki = 8300 nM T60693 C0RI4V 13298444 Ki = 61 nM T60693 CNJ1Q6 13559325 Ki = 10.1 nM T60693 C06ADH 13599612 Ki > 10000 nM T60693 CAK28N 13787553 Ki = 7.7 nM T60693 C2UQX9 13911081 Ki = 3.7 nM T60693 C7M4BP 13911085 Ki = 816 nM T60693 C9C5TY 14570180 Ki > 1000 nM T60693 C0UX9N 14570184 Ki = 2325 nM T60693 C23ZPH 14810949 IC50 = 102 nM T60693 CPJA56 14810957 IC50 = 260 nM T60693 C4G3ZF 14933784 IC50 = 0.39 nM T60693 CK5I1M 14933785 IC50 = 6 nM T60693 CPHW81 15033953 Ki = 20 nM T60693 CD56LF 15033955 Ki = 820 nM T60693 C75DUO 15123215 IC50 = 69 nM T60693 CNX8R5 15123216 IC50 = 0.88 nM T60693 CWP7F4 15123217 IC50 = 6.3 nM T60693 C9YW7A 15123218 IC50 = 15 nM T60693 C8RN0Z 15123220 IC50 = 29 nM T60693 C6MV4I 15123221 IC50 = 4.7 nM T60693 CHZ79J 15123222 IC50 = 1020 nM T60693 CQP65B 15123223 IC50 = 0.12 nM T60693 C97TSQ 15123224 IC50 = 690 nM T60693 CFV78H 15123226 IC50 = 550 nM T60693 C4ZK5U 15123234 IC50 > 10000 nM T60693 CIL30V 15123235 IC50 > 10000 nM T60693 C0MUJ3 15123237 IC50 = 590 nM T60693 C5WI6C 15123238 IC50 = 970 nM T60693 CMR2Z0 15123240 IC50 = 2000 nM T60693 CW9NG6 15123248 IC50 = 46 nM T60693 C69EXU 15123249 IC50 = 120 nM T60693 CCGA13 15123251 IC50 = 5 nM T60693 CS5QJ0 15123254 IC50 = 250 nM T60693 C06NJO 15123255 IC50 = 1200 nM T60693 CI7O6D 15123272 IC50 = 57 nM T60693 CH2Q9J 15123276 IC50 > 10000 nM T60693 C1GDR7 15123277 IC50 = 2200 nM T60693 CK9PA4 15123278 IC50 > 10000 nM T60693 CF27TQ 15384274 Ki > 10000 nM T60693 CUND10 15407235 IC50 = 8759 nM T60693 CAW1M2 15512228 Ki = 25.12 nM T60693 C30CHU 15512229 Ki = 19.95 nM T60693 C9B5OD 15512233 Ki = 158.49 nM T60693 CX6H8V 15512234 Ki = 50.12 nM T60693 CC5X0L 15512235 Ki = 19.95 nM T60693 C53KRM 15512237 Ki = 12.59 nM T60693 CLA5K8 15512238 Ki = 79.43 nM T60693 CSX74V 15512240 Ki = 79.43 nM T60693 CET25R 15512241 Ki = 199.53 nM T60693 C7CNY1 15512243 Ki = 63.1 nM T60693 CZA4J8 15541261 Ki = 137 nM T60693 CV46FB 15546394 Ki = 0.091 nM T60693 CRM01L 15548354 Ki = 0.4266 nM T60693 C1DB3A 15548355 Ki = 0.69 nM T60693 C7Q3JW 15560576 Ki = 116 nM T60693 C7L6UQ 15645955 IC50 = 15 nM T60693 C6DLW3 15645956 IC50 = 10 nM T60693 CIS8G3 15645957 IC50 = 6.9 nM T60693 C3R4XO 15645958 IC50 = 60 nM T60693 C1Z4QY 15645959 IC50 = 2900 nM T60693 CV04HA 15645960 IC50 = 0.42 nM T60693 CC2VB5 15645961 IC50 > 10000 nM T60693 C2DO5R 15645962 IC50 > 10000 nM T60693 CF3M4T 15645964 IC50 = 3.5 nM T60693 COA3P2 15645965 IC50 = 300 nM T60693 CM0NH8 15645966 IC50 > 10000 nM T60693 CJC1S7 15645967 IC50 = 450 nM T60693 CXN5K2 15645974 IC50 = 0.04 nM T60693 CKP3V6 15645975 IC50 = 1.2 nM T60693 CS1B5Q 15645978 IC50 = 0.34 nM T60693 C20LMY 15645979 IC50 = 0.34 nM T60693 CREN90 15645980 IC50 = 4 nM T60693 CVRI70 15645981 IC50 = 0.28 nM T60693 C9TYD1 15923664 Ki > 100000 nM T60693 C75LOT 15934554 Ki = 110 nM T60693 C6DW5M 15982528 IC50 > 10000 nM T60693 C7Z8OD 15982529 IC50 = 97 nM T60693 CV1G7O 15982660 IC50 = 480 nM T60693 CG3L8Z 15982661 IC50 = 100 nM T60693 CN64AP 15982791 IC50 = 220 nM T60693 CJ6W1T 15982933 IC50 > 10000 nM T60693 CV3TQ9 16006949 Ki = 1.8 nM T60693 CA5GL7 16007142 Ki = 2780 nM T60693 CD3BS8 16007286 EC50 = 0.75 nM T60693 CK3QD9 16039356 Ki = 4910 nM T60693 C3XA7E 16048783 Ki = 11 nM T60693 CDV05T 16048784 Ki = 2.7 nM T60693 C3O4HX 16048863 Ki = 3.3 nM T60693 CPV60X 16048864 Ki = 3.2 nM T60693 CFZI17 16048866 Ki = 0.38 nM T60693 CNDV23 16048867 Ki = 0.063 nM T60693 C9SCH7 16048936 Ki = 19 nM T60693 C6A5UL 16048937 Ki = 2.4 nM T60693 C3PO9S 16048938 Ki = 0.2 nM T60693 CJ6LM3 16048939 Ki = 1.9 nM T60693 CUQ16Z 16048940 Ki = 0.18 nM T60693 CG71OP 16048941 Ki = 2.2 nM T60693 CP23YA 16049012 Ki = 2.4 nM T60693 CQK63V 16051935 IC50 = 217 nM T60693 C6LFA8 16059781 Ki = 540 nM T60693 CSK23U 16083041 Ki = 0.35 nM T60693 CR0S9Y 16087270 IC50 = 0.003 nM T60693 CSB90O 16087271 Ki = 4.94 nM T60693 C75QOB 16087272 IC50 = 3.45 nM T60693 CP5B0A 16087273 Ki = 3.69 nM T60693 CK8C3L 16087274 Ki = 1 nM T60693 CBW82T 16087275 IC50 = 0.29 nM T60693 CFZ95P 16087276 Ki = 25.2 nM T60693 C48WDR 16087277 Ki = 7.51 nM T60693 C7V4ZB 16087278 Ki = 33.5 nM T60693 C8X5HT 16087279 Ki = 41.5 nM T60693 CE7G1T 16087280 Ki = 13.1 nM T60693 C4B1NT 16087283 IC50 = 0.006 nM T60693 CU1J5C 16087284 IC50 = 0.59 nM T60693 CU15KC 16087285 IC50 = 0.44 nM T60693 C30MPR 16087286 IC50 = 0.34 nM T60693 CITF65 16087287 IC50 = 1.87 nM T60693 CN5KV0 16087288 Ki = 21.5 nM T60693 C4FW9H 16087289 Ki = 25.9 nM T60693 C2OVH1 16087290 Ki = 2.59 nM T60693 CLYD13 16094317 Ki = 1400 nM T60693 C8W1BR 16094318 Ki = 440 nM T60693 C3S7GV 16094319 Ki = 100 nM T60693 CR71BM 16094320 Ki = 35 nM T60693 C6VS7F 16094321 Ki = 520 nM T60693 CV1P4O 16094322 Ki = 69 nM T60693 CZ4V9I 16094342 Ki = 430 nM T60693 CO8T5W 16094343 IC50 = 1.2 nM T60693 C0I9GV 16094344 Ki = 65 nM T60693 C21JYZ 16094345 Ki = 16 nM T60693 CEDY75 16094347 Ki = 520 nM T60693 C3SZX8 16094366 Ki = 540 nM T60693 C5RGW0 16094367 IC50 = 15 nM T60693 CB46JH 16094368 Ki = 130 nM T60693 CCLO14 16094369 Ki = 300 nM T60693 CUN6E1 16094370 IC50 = 10 nM T60693 C9QI4H 16094371 Ki = 83 nM T60693 C90BWG 16094372 Ki = 280 nM T60693 CTY5V3 16094373 IC50 = 9.4 nM T60693 C23KIF 16094374 Ki = 56 nM T60693 C48EXZ 16094375 Ki = 270 nM T60693 C9UR3E 16094377 Ki = 140 nM T60693 COG76W 16094378 Ki = 24 nM T60693 CBS04I 16094379 Ki = 33 nM T60693 C7AQL2 16094380 Ki = 980 nM T60693 CMJ5H3 16094381 Ki = 230 nM T60693 CL1A7O 16094383 Ki = 390 nM T60693 CKS40Z 16094384 Ki = 400 nM T60693 C5WZF1 16094386 Ki = 430 nM T60693 CYP92H 16094387 Ki = 120 nM T60693 CGRX31 16094388 IC50 = 6.6 nM T60693 CO4Z1K 16094389 Ki = 38 nM T60693 CH23IJ 16094390 IC50 = 36 nM T60693 C0N6ID 16094393 Ki = 620 nM T60693 CS8L3K 16094394 IC50 = 99 nM T60693 CX87TS 16094397 Ki = 460 nM T60693 C4RIZ1 16094408 Ki = 430 nM T60693 C4D1UF 16094410 Ki = 130 nM T60693 C7V1YT 16094411 Ki = 57 nM T60693 CUA2L0 16094413 Ki = 540 nM T60693 C3AMW5 16094414 IC50 = 8.4 nM T60693 C6J0YV 16094415 Ki = 950 nM T60693 CX4K0L 16094416 Ki = 420 nM T60693 CR7AS8 16094419 Ki = 3700 nM T60693 CK98PS 16094420 IC50 = 3.2 nM T60693 C9AJK7 16094421 IC50 = 2.4 nM T60693 CI2XK6 16094424 IC50 = 2.3 nM T60693 C6GL2A 16094425 IC50 = 16 nM T60693 CO4M3A 16094426 IC50 = 1.2 nM T60693 C1JBM6 16094428 IC50 = 50 nM T60693 CK7N1Y 16094430 IC50 = 20 nM T60693 C8P6JV 16095099 Ki = 7 nM T60693 CB90WO 16358672 Ki = 707.95 nM T60693 C0XT4U 16445678 Ki = 1100 nM T60693 CC02SB 16446593 Ki = 512.86 nM T60693 CZ2IS9 16660294 Ki > 10000 nM T60693 C08RXS 16665915 Ki = 820 nM T60693 CS9FW1 16665917 Ki = 180 nM T60693 C1LX0I 16665918 Ki = 1890 nM T60693 CCF0J7 16720551 Ki = 1.4 nM T60693 C0ACW1 16720553 Ki = 14 nM T60693 CG6OD7 16720646 Ki = 1 nM T60693 CC4N5P 16720648 Ki = 1.9 nM T60693 CFI67Y 16720649 Ki = 2.2 nM T60693 C8GOL2 16720650 Ki = 0.14 nM T60693 CB9MZ5 16720745 Ki = 0.64 nM T60693 CAY72B 16720746 Ki = 390 nM T60693 CO84NU 16720747 Ki = 89 nM T60693 CG62NU 16720749 Ki = 0.07 nM T60693 C8SOD5 16735664 Ki = 153 nM T60693 C4ORI6 16739256 Ki = 938 nM T60693 C1MFJ2 16747695 Ki = 174 nM T60693 C5UGV2 16748227 Ki = 40 nM T60693 CO0XL6 16748228 Ki = 3400 nM T60693 CNEX42 16748229 Ki = 300 nM T60693 CN4JB2 16748352 Ki = 180 nM T60693 CJX60K 16748353 Ki = 125 nM T60693 C5W1UD 16748354 Ki = 910 nM T60693 C9ZD4O 16748355 Ki = 3.7 nM T60693 C9TC3L 16748356 Ki = 420 nM T60693 C68VNE 16748478 Ki = 25 nM T60693 C6QMJ9 16756731 Ki = 3830 nM T60693 C4AEU1 16756734 Ki = 245 nM T60693 C9D5RB 16756735 Ki = 690 nM T60693 C2BG6Z 16756840 Ki = 184 nM T60693 C0Q2OC 16756841 Ki = 235 nM T60693 C6NF5U 16756953 Ki = 150 nM T60693 CS26LH 16757050 Ki = 4 nM T60693 CFS39T 16757147 Ki = 15 nM T60693 CJY27L 17798965 Ki = 1.3 nM T60693 C6IW7Z 17798971 Ki = 6.3 nM T60693 CIQ2R5 17798973 Ki = 2.9 nM T60693 CX91VE 17798974 Ki = 5 nM T60693 CGB04N 17798976 Ki = 75 nM T60693 CYJ06B 17798978 Ki = 3.6 nM T60693 CJNQ89 17925232 Ki = 24 nM T60693 C4UYA0 18607197 Ki = 69 nM T60693 C1Y9FT 18782352 Ki = 33.5 nM T60693 CYUG80 18782376 Ki = 66.5 nM T60693 C46DPT 18782378 Ki = 94.5 nM T60693 C73DWV 18782384 Ki = 203 nM T60693 CL17VG 18955362 IC50 = 3.5 nM T60693 C61OBX 19881394 Ki = 12.6 nM T60693 C7T8JC 19958494 Ki > 10000 nM T60693 C6LI5E 19958507 Ki > 10000 nM T60693 C5BE7T 20345831 IC50 = 18600 nM T60693 C3I8EH 20642899 Ki = 4800 nM T60693 C94FLX 20833183 IC50 = 41.1 nM T60693 C4HAP8 20900833 Ki = 9772.37 nM T60693 CIOT38 20968607 IC50 > 32000 nM T60693 CBX5O7 21074158 Ki = 29 nM T60693 C3T5HF 21509921 Ki = 1995.26 nM T60693 C72JWU 21589299 EC50 = 3.34 nM T60693 CBN84K 22065997 Ki > 10000 nM T60693 CS24KZ 22213385 Ki = 21.6 nM T60693 CHAI36 22272877 IC50 = 120 nM T60693 CX3JY4 22273116 IC50 = 60 nM T60693 C6IGK7 22475272 Ki = 3284 nM T60693 CTDP73 22509672 Ki = 363.08 nM T60693 C0ESJ4 22509676 Ki = 645.65 nM T60693 C1W7MX 22522554 IC50 = 4320 nM T60693 C90UPB 22553442 IC50 = 1300 nM T60693 C8DF5U 22558157 Ki = 15.13 nM T60693 C1R5PV 22562132 Ki > 2000 nM T60693 CJ8OB0 22562135 Ki > 2000 nM T60693 C0GKU4 22562137 Ki = 70.04 nM T60693 C4ZL2N 22573197 Ki = 22 nM T60693 C5YZ9U 22573205 Ki = 0.34 nM T60693 CO84SM 22573206 Ki = 2 nM T60693 CXE34L 22573216 Ki = 1900 nM T60693 CKI1O3 22573217 Ki = 0.72 nM T60693 CR1PV4 22573223 Ki = 2.6 nM T60693 CD4C5N 22729898 Ki = 95 nM T60693 CX3O6L 22729907 Ki = 347 nM T60693 C7OL1R 22729922 Ki = 150 nM T60693 CA28YU 22729923 Ki = 440 nM T60693 CSP6M3 22810742 Ki = 363 nM T60693 CG60MD 22816300 Ki = 589 nM T60693 CL7X2U 23383556 Ki = 10 nM T60693 COHN67 23383564 Ki = 30 nM T60693 CBW20U 23435898 IC50 > 10000 nM T60693 C46ZSX 23542099 IC50 = 240 nM T60693 C8ZD9W 23567095 Ki = 14.7 nM T60693 C9NI1F 23567109 Ki = 0.8 nM T60693 CZQP15 23567112 Ki = 1.3 nM T60693 C10UWF 23567114 Ki = 3.6 nM T60693 CIPX37 23567116 Ki = 4.5 nM T60693 CCT6R7 23567120 Ki = 3.9 nM T60693 CNH40T 23567127 Ki = 2.4 nM T60693 C1Y8CH 23567131 Ki = 3.3 nM T60693 CJD8Q6 23567134 Ki = 99 nM T60693 C54SJG 23567138 Ki = 1.3 nM T60693 C3K6HV 23594220 Ki = 5.9 nM T60693 CVBM54 23594222 Ki = 47 nM T60693 CXC6E3 23594223 Ki = 5.9 nM T60693 CQ93SH 23594225 Ki = 0.8 nM T60693 CC5E7N 23594227 EC50 = 1 nM T60693 CG3M5J 23594230 Ki = 2.8 nM T60693 C5L8ZA 23594232 Ki = 1.7 nM T60693 C08XMZ 23594241 Ki = 1.3 nM T60693 C0D5AC 23594243 Ki = 2.7 nM T60693 C4JGI8 23594247 Ki = 1.7 nM T60693 CXN07F 23661598 Ki = 310 nM T60693 CA9W3S 23726012 Ki = 0.033 nM T60693 CO5YP3 23986637 Ki = 0.18 nM T60693 CY0UD4 24180494 Ki = 79 nM T60693 CB9MC8 24735827 Ki = 321 nM T60693 C84JOU 24754997 Ki = 187.97 nM T60693 CWP85S 24776395 Ki = 557 nM T60693 CVD48X 24776396 Ki = 412 nM T60693 C3WDL8 24776397 Ki = 103 nM T60693 CXL4R0 24776398 Ki = 178 nM T60693 CR9I1S 24776399 Ki = 3600 nM T60693 CQDJ35 24776400 Ki = 1150 nM T60693 C6CX0Z 24776401 Ki = 928 nM T60693 CJH18I 24776402 Ki = 123 nM T60693 C27SGI 24776403 Ki = 1920 nM T60693 CV5IG2 24776404 Ki = 97 nM T60693 CQ70IW 24776405 Ki = 190 nM T60693 CQ2P5J 24776406 Ki = 1104 nM T60693 CYIV42 24776407 Ki = 3827 nM T60693 CWB06Z 24776408 Ki = 3977 nM T60693 C36WQO 24776409 Ki = 3844 nM T60693 CUP2C6 24776410 Ki = 3641 nM T60693 CC3W7E 24776411 Ki > 10000 nM T60693 C3N6GE 24776412 Ki > 10000 nM T60693 C2M6BR 24776413 Ki > 10000 nM T60693 CS01RL 24800107 Ki = 15 nM T60693 CL2WB0 24800108 Ki = 23.1 nM T60693 CFIS62 24822296 Ki = 0.29 nM T60693 CB4S7U 24822297 Ki = 0.4 nM T60693 CC06ON 24822298 Ki = 0.79 nM T60693 C30GOT 24822299 Ki = 0.043 nM T60693 C2B3EM 24822300 Ki = 0.45 nM T60693 C1JRM9 24822458 Ki = 0.42 nM T60693 C5VYZ2 24822459 Ki = 2.74 nM T60693 CIC3L7 24822460 Ki = 0.51 nM T60693 C7O9BN 24822461 Ki = 4.5 nM T60693 C13MJI 24822630 Ki = 0.1 nM T60693 CJK3I4 24822631 Ki = 0.72 nM T60693 CW2B0R 24822632 Ki = 0.28 nM T60693 CRT19I 24822633 Ki = 2.41 nM T60693 CN6JX5 24822634 Ki = 0.73 nM T60693 CCKO91 24822798 Ki = 0.39 nM T60693 CPN52E 24822799 Ki = 0.24 nM T60693 C58EYR 24822801 Ki = 150.61 nM T60693 CBYW42 24822802 Ki = 0.09 nM T60693 CAK7O3 24822964 Ki = 0.43 nM T60693 C6R3AE 24822965 Ki = 1.2 nM T60693 CYQ27T 24824634 Ki = 2.03 nM T60693 C6TWH4 24824635 Ki = 0.23 nM T60693 CBPQ24 24824636 Ki = 0.06 nM T60693 CCY7A8 24824637 Ki = 0.16 nM T60693 C9G0CI 24824638 Ki = 0.78 nM T60693 CT0PG3 24828463 Ki = 11600 nM T60693 CTZ0S2 24829369 Ki = 7430 nM T60693 CDC91N 24839550 Ki = 2454.71 nM T60693 CI4W6P 24854099 Ki = 230 nM T60693 CV6NW8 24854100 Ki = 550 nM T60693 C5ZCJ9 24854101 Ki = 900 nM T60693 CZM9I7 24854102 Ki = 800 nM T60693 CO7LG3 24854177 Ki = 570 nM T60693 C75WFT 24854178 Ki = 410 nM T60693 CC5KH6 24854179 Ki = 5490 nM T60693 CL06MB 24854180 Ki = 70 nM T60693 C7ED1M 24854260 Ki = 80 nM T60693 C0I4KH 24854261 Ki = 2010 nM T60693 C2ZUH5 24854262 Ki = 260 nM T60693 CS3JT4 24854263 Ki = 1400 nM T60693 C53SWQ 24854264 Ki = 1410 nM T60693 C9O5NZ 24857819 IC50 = 120 nM T60693 CN0T1F 24857820 IC50 = 170 nM T60693 CECI63 24858447 Ki > 10000 nM T60693 CM80JI 24863522 EC50 = 2000 nM T60693 CRUQ41 24863611 IC50 > 10000 nM T60693 CIJ83R 24873473 Ki = 0.22 nM T60693 CK61ND 24886211 Ki > 10000 nM T60693 CDR3T2 24886213 Ki > 10000 nM T60693 CNQ6I4 24894028 IC50 > 10000 nM T60693 C71NXE 24970312 EC50 = 1300 nM T60693 CT09XK 24978531 IC50 = 1770 nM T60693 CIY83H 24995848 Ki = 17.4 nM T60693 CDLW86 25001412 Ki = 316.23 nM T60693 CA76KJ 25067046 EC50 = 6300 nM T60693 CWU10S 25071953 EC50 = 2000 nM T60693 CHR36S 25074770 Ki = 10 nM T60693 CU4C8F 25077980 Ki = 10 nM T60693 CUO63Q 25129091 Ki = 2000 nM T60693 CQ36GH 25129435 Ki = 520 nM T60693 C60PHW 25169521 EC50 = 0.11 nM T60693 CV3Y7O 25169522 EC50 = 0.43 nM T60693 CG6UT3 25181466 Ki = 0.55 nM T60693 CF6RA5 25190572 Ki = 506 nM T60693 CPK5D7 25190573 Ki = 1342 nM T60693 CON62K 25190574 Ki = 773 nM T60693 C6S3WN 25190575 Ki = 633 nM T60693 CF15AH 25190576 Ki = 1846 nM T60693 CBN1Q0 25190577 Ki = 2316 nM T60693 CKB72D 25190578 Ki = 1268 nM T60693 CZR78G 25190579 Ki = 694 nM T60693 CF2JK0 25190580 Ki = 81010 nM T60693 CE4R2X 25190581 Ki = 46515 nM T60693 CYC6S0 25190582 Ki = 2274 nM T60693 CE61QB 25190583 Ki = 1747 nM T60693 C9V8MS 25190584 Ki = 1830 nM T60693 C3UV5M 25190585 Ki = 852 nM T60693 CKFI42 25190586 Ki = 497 nM T60693 C5UQX3 25190587 Ki = 469 nM T60693 C5J2WE 25190588 Ki = 247 nM T60693 CX84WI 25190589 Ki = 224 nM T60693 C5RUI9 25190590 Ki = 320 nM T60693 CQY69C 25190591 Ki = 1014 nM T60693 C8SEQ2 25190592 Ki = 674 nM T60693 C5BS7N 25190593 Ki = 165 nM T60693 CE19OU 25190594 Ki = 238 nM T60693 CP5ID6 25190595 Ki = 271 nM T60693 CO8E4G 25190596 Ki = 64 nM T60693 CX87HD 25190597 Ki = 279 nM T60693 CY6CV1 25190598 Ki = 52 nM T60693 CW5UP9 25190599 Ki = 68 nM T60693 C1C8VK 25190600 Ki = 54 nM T60693 CL7Q2F 25190601 Ki = 40 nM T60693 CD0H5U 25190602 Ki = 25 nM T60693 C8OWC0 25190603 Ki = 29 nM T60693 CH06YU 25190604 Ki = 13 nM T60693 CEJ25L 25190605 Ki = 8 nM T60693 CXD5R8 25190606 Ki = 56 nM T60693 CU6W8O 25190607 Ki = 1392 nM T60693 CWJB54 25190608 Ki = 56 nM T60693 CMHS48 25190609 Ki = 655 nM T60693 CBL9S4 25190610 Ki = 48 nM T60693 CZ8Y6L 25190611 Ki = 39 nM T60693 CL9SN6 25190612 Ki = 68 nM T60693 C1MGY3 25190613 Ki = 49 nM T60693 CB1G6M 25190614 Ki = 33 nM T60693 CJLH27 25190615 Ki = 45 nM T60693 COE65V 25190616 Ki = 208 nM T60693 C30VGA 25190617 Ki = 45 nM T60693 CO7IV2 25190618 Ki = 174 nM T60693 C8Q7WV 25190619 Ki = 65 nM T60693 C0G4RJ 25190620 Ki = 86 nM T60693 C7X4IV 25190621 Ki = 169 nM T60693 CXG8O3 25190622 Ki = 138 nM T60693 CD5F6A 25190623 Ki = 82 nM T60693 CFUD47 25190624 Ki = 540 nM T60693 C15LIW 25190625 Ki = 26 nM T60693 C3LEW8 25190626 Ki = 151 nM T60693 CIDV61 25190627 Ki = 11 nM T60693 CAGS39 25190628 Ki = 14 nM T60693 CDS2E6 25190629 Ki = 25 nM T60693 CPW19O 25190630 Ki = 158 nM T60693 C0SBV7 25207946 Ki = 352 nM T60693 C21OJF 25207948 Ki = 43 nM T60693 C0P6CS 25207950 Ki = 72 nM T60693 CN9I8E 25208095 Ki = 25 nM T60693 C5OA1N 25208097 EC50 = 8.4 nM T60693 C59IKP 25208099 Ki = 10 nM T60693 C9BJD3 25232367 Ki = 77.23 nM T60693 CK0F7G 25232539 Ki = 5.42 nM T60693 CGLZ15 25232540 EC50 = 28.8 nM T60693 CHG71D 25232541 Ki = 26.45 nM T60693 CGH3W8 25232542 Ki = 9.84 nM T60693 C8E0RL 25232543 Ki = 5.04 nM T60693 CE6JP0 25232724 Ki = 0.57 nM T60693 C0OU5Y 25232725 Ki = 608.76 nM T60693 C3LHO0 25232727 Ki = 222.58 nM T60693 CO74DE 25233078 Ki = 1.81 nM T60693 CJS1L7 25233081 Ki = 65.26 nM T60693 C1INO6 25233083 Ki = 1.58 nM T60693 C83AVG 25233258 Ki = 19.56 nM T60693 CKL48U 25256790 Ki = 25.5 nM T60693 C4CP2G 25256965 EC50 = 0.079 nM T60693 CY54AO 25256967 Ki = 0.59 nM T60693 CLK31Y 25256969 Ki = 1.1 nM T60693 CYSU80 25257195 Ki = 0.27 nM T60693 C9NC3W 25257431 Ki = 4.3 nM T60693 C2GH4L 25257432 Ki = 52 nM T60693 C0EC4L 25257433 Ki = 36 nM T60693 C47YRW 25259489 Ki = 0.3 nM T60693 CZK9Q8 25259490 EC50 = 0.12 nM T60693 C5R6YL 25259957 Ki = 0.26 nM T60693 CGO9W2 25260181 EC50 = 0.78 nM T60693 C7XY9W 25270622 IC50 > 10000 nM T60693 CBD0K9 25270623 IC50 > 10000 nM T60693 CL2Z7J 42629117 Ki = 752 nM T60693 CJ3X7R 42636619 EC50 = 35 nM T60693 C0K9TG 44138064 Ki = 0.81 nM T60693 C15NFW 44138152 Ki = 450 nM T60693 CL57VS 44143431 IC50 = 530 nM T60693 C6GDL8 44143433 IC50 = 160 nM T60693 CPQ25W 44181744 Ki = 518 nM T60693 CX4D3R 44188273 Ki = 1.66 nM T60693 C2XE7Y 44189733 IC50 = 10000 nM T60693 CGA8R1 44189735 IC50 = 6800 nM T60693 C50FOG 44189834 IC50 = 11000 nM T60693 C2AV1K 44190762 IC50 = 3480 nM T60693 CCV87B 44235260 Ki = 5120 nM T60693 CV2NB5 44235261 Ki = 1190 nM T60693 C0X3VW 44235262 Ki = 2550 nM T60693 C2HM9V 44235488 EC50 = 62.1 nM T60693 CCO7H6 44235489 Ki = 3810 nM T60693 CW7NH4 44235490 EC50 = 67.1 nM T60693 C6NIL8 44235491 Ki = 1520 nM T60693 CG9QD7 44240971 Ki = 1.8 nM T60693 CR61KZ 44240972 EC50 = 2.6 nM T60693 C0AL2R 44241022 Ki = 2.6 nM T60693 CK5T9S 44241023 Ki = 1.7 nM T60693 C6D0HY 44241024 Ki = 3 nM T60693 C5G6DN 44241123 Ki = 1.5 nM T60693 CM48UY 44244681 Ki = 140 nM T60693 CC63QX 44247589 Ki = 1610 nM T60693 CJW3P2 44254063 Ki = 390 nM T60693 C9SQ8D 44254859 Ki = 1600 nM T60693 CVCP62 44254956 Ki = 890 nM T60693 C8HI7P 44256416 IC50 = 6.68 nM T60693 C4PG9V 44269757 IC50 = 25 nM T60693 C0YTQ7 44269766 IC50 = 2450 nM T60693 CW75BD 44269767 IC50 = 2.3 nM T60693 C2FDR9 44269802 IC50 = 550 nM T60693 C32OQJ 44269803 IC50 = 1760 nM T60693 CY61IX 44269822 IC50 = 41 nM T60693 CW7C4R 44269855 IC50 = 1400 nM T60693 CUH74K 44269856 IC50 = 8.4 nM T60693 CMIZ34 44269859 IC50 = 33 nM T60693 CG93NF 44269868 IC50 = 330 nM T60693 CE26RM 44269871 IC50 = 94 nM T60693 C35VDR 44269872 IC50 = 465 nM T60693 C6Y8IM 44269891 IC50 = 82 nM T60693 C3X2ID 44269895 IC50 = 94 nM T60693 CW4PS6 44269900 IC50 > 10000 nM T60693 CM62ZD 44269901 IC50 = 14 nM T60693 C6T9WO 44269902 IC50 = 56 nM T60693 CQ2W3Z 44269927 IC50 = 9.6 nM T60693 C2CAI8 44269932 IC50 = 420 nM T60693 CJQI23 44269933 IC50 = 320 nM T60693 C8AMT3 44269936 IC50 = 22 nM T60693 C9H0AG 44269950 IC50 = 7.6 nM T60693 CQ20KW 44269951 IC50 = 38 nM T60693 C89YQU 44269952 IC50 = 13 nM T60693 C0H4SW 44269967 IC50 = 6.9 nM T60693 CA2L4V 44269968 IC50 > 1000 nM T60693 CZ49TF 44269969 IC50 = 57 nM T60693 CTRE60 44269980 IC50 = 3080 nM T60693 CIFJ07 44269988 IC50 = 9.8 nM T60693 CWU8M4 44269994 IC50 = 5.5 nM T60693 CAG2N4 44270012 IC50 = 53 nM T60693 C2CEN5 44273397 EC50 = 1.1 nM T60693 CW6P4Y 44276782 Ki > 10000 nM T60693 CC2OD4 44278111 Ki > 10000 nM T60693 CRMA84 44278114 Ki > 10000 nM T60693 CF0Y4M 44278115 Ki > 10000 nM T60693 CUS04C 44279592 Ki = 0.87 nM T60693 CL70JN 44279594 Ki = 1.28 nM T60693 C3AYK9 44279686 EC50 = 0.1 nM T60693 C9STZ5 44279699 EC50 = 0.04 nM T60693 CX9KP8 44284742 Ki = 110 nM T60693 CWKT78 44285029 Ki = 250 nM T60693 CQ15BW 44285070 Ki > 500 nM T60693 CN7V6X 44286598 Ki = 303 nM T60693 CV46BG 44286647 Ki = 130 nM T60693 C69JKC 44286719 Ki = 543 nM T60693 CY9PS5 44286720 Ki = 39.5 nM T60693 C6QZ4H 44286867 IC50 = 1.53 nM T60693 C6NQ5U 44286870 Ki > 1000 nM T60693 C6SJY9 44286875 IC50 = 501 nM T60693 C4CYJ1 44286876 IC50 = 26 nM T60693 C41IRN 44286883 Ki > 1000 nM T60693 CNOB73 44286884 Ki > 1000 nM T60693 C7SZ0Y 44286885 Ki = 511 nM T60693 C3JRH1 44286895 IC50 = 184 nM T60693 CS54YC 44287020 IC50 = 40.5 nM T60693 CHU57Z 44287142 Ki = 310 nM T60693 C39XJE 44287143 Ki > 1000 nM T60693 C2Y3MA 44287144 Ki > 1000 nM T60693 CRO32K 44287168 Ki > 1000 nM T60693 C09XZL 44287189 Ki = 109 nM T60693 CW9TN6 44287225 IC50 = 9.98 nM T60693 C8U5QT 44287236 Ki = 481 nM T60693 C0RE2U 44287369 Ki = 405 nM T60693 CL6K5U 44287383 Ki > 1000 nM T60693 CQ46MS 44287394 Ki > 1000 nM T60693 CQU8Z1 44287414 Ki = 480 nM T60693 C7M2FV 44287415 Ki > 1000 nM T60693 C1RE2J 44287486 Ki = 530 nM T60693 C97UNH 44287487 Ki = 194 nM T60693 CE8WC0 44288497 Ki = 53 nM T60693 C12VDA 44288499 Ki = 16 nM T60693 C6THR2 44288512 Ki = 12 nM T60693 CJH12A 44288798 Ki = 333 nM T60693 CVJ9M3 44288802 Ki = 28000 nM T60693 CE57CX 44288830 Ki = 37000 nM T60693 CV26NK 44288832 Ki = 17 nM T60693 C9J6GY 44288940 Ki = 94 nM T60693 C7JX2K 44288942 Ki = 146 nM T60693 C8K9AW 44288968 Ki = 2000 nM T60693 CY7S9C 44289066 Ki = 180 nM T60693 CRUP26 44289068 Ki = 180 nM T60693 C5MU4H 44289172 Ki = 25000 nM T60693 C0S9PH 44289174 Ki = 8100 nM T60693 CN46EU 44289190 Ki = 7 nM T60693 C6JH4F 44289193 Ki = 261 nM T60693 C3BD9K 44289212 Ki = 154 nM T60693 C2YV1Z 44289252 Ki = 17 nM T60693 C5WE4Y 44292142 IC50 > 10000 nM T60693 CE3YS4 44292200 IC50 = 89 nM T60693 C0VR9X 44292280 IC50 = 9000 nM T60693 CIEU38 44292281 IC50 = 9290 nM T60693 CARS41 44292403 IC50 > 10000 nM T60693 C2ST7W 44292414 IC50 = 2730 nM T60693 C3KYZ5 44292426 IC50 > 10000 nM T60693 C2ET5R 44292437 IC50 > 10000 nM T60693 C6MQ8U 44295810 Ki = 0.006 nM T60693 C9AF6B 44297435 Ki = 2.3 nM T60693 CNP5W1 44297519 Ki = 271 nM T60693 C9UY4E 44297697 Ki = 987 nM T60693 C8F1ST 44297727 Ki = 227 nM T60693 C4YG5R 44298841 Ki = 13 nM T60693 CF8YG9 44299258 Ki = 220 nM T60693 C7ZYM4 44299404 Ki > 350 nM T60693 CTB24D 44299841 Ki = 270 nM T60693 CT6HW3 44300146 Ki = 0.47 nM T60693 C9IL2D 44301524 Ki = 74.1 nM T60693 CG6JI1 44301701 EC50 = 1.7 nM T60693 C26CLF 44302821 IC50 = 2.4 nM T60693 CNI7U6 44302972 IC50 = 2.2 nM T60693 CL6I9X 44302973 IC50 = 19.5 nM T60693 CB2H7L 44302988 IC50 = 5.7 nM T60693 C28OYR 44302993 IC50 = 34.2 nM T60693 CGV70Q 44302996 IC50 = 1494 nM T60693 C3RX4Q 44303011 IC50 = 524 nM T60693 C23GUZ 44303030 IC50 = 31.9 nM T60693 CWM93O 44303041 IC50 = 49.4 nM T60693 CI3E0C 44303074 IC50 = 1177 nM T60693 CL2D8J 44303092 IC50 = 271 nM T60693 C4VN8H 44303094 IC50 = 22.5 nM T60693 C2RTS0 44303112 IC50 = 3.44 nM T60693 CGS81I 44303376 IC50 = 5.5 nM T60693 CXN7F0 44303379 IC50 = 34.8 nM T60693 CICN21 44303386 IC50 = 3.4 nM T60693 C2L9UZ 44303682 IC50 = 5.3 nM T60693 C1CI7Y 44303692 IC50 = 79.3 nM T60693 CY0HT8 44306645 IC50 = 14.3 nM T60693 CWT5Q7 44306866 Ki = 0.35 nM T60693 CXG6D2 44306867 Ki = 0.15 nM T60693 COIN83 44306936 IC50 = 1183 nM T60693 CSA9Y2 44306943 IC50 = 0.06 nM T60693 C1IBV3 44306952 IC50 = 2.6 nM T60693 C62VYD 44307037 IC50 = 13000 nM T60693 C3ZQR0 44307038 IC50 = 189 nM T60693 CU73AD 44307039 IC50 > 2000 nM T60693 CWY7L4 44307076 IC50 = 301 nM T60693 CMU1T6 44307167 IC50 = 45.5 nM T60693 CH0YD7 44307168 IC50 = 85.5 nM T60693 C4GV6L 44307169 IC50 = 738 nM T60693 C2CA8S 44307170 IC50 = 125 nM T60693 CB37KT 44307185 IC50 = 20 nM T60693 C0X3HL 44307191 Ki = 0.23 nM T60693 CU93BT 44307213 IC50 = 152 nM T60693 C4E3GT 44307234 IC50 = 17.4 nM T60693 CBO97V 44307317 IC50 = 4.9 nM T60693 COS3X0 44307318 IC50 = 2.3 nM T60693 CB1P0W 44307319 IC50 = 1.07 nM T60693 C0E5ZU 44307320 IC50 = 24 nM T60693 CG4JZ5 44307987 IC50 = 3.8 nM T60693 C9S2IM 44308032 IC50 = 3.4 nM T60693 C0GJT5 44311043 Ki = 34 nM T60693 C2GE8X 44311351 Ki = 88 nM T60693 CV9X4Q 44311893 Ki = 0.17 nM T60693 CLX5V8 44312109 Ki = 0.12 nM T60693 C9J7BL 44320576 Ki = 0.096 nM T60693 CT6E9J 44320593 Ki = 0.086 nM T60693 CM0G8A 44324324 Ki = 94 nM T60693 CALT96 44324339 Ki = 65 nM T60693 C2Y4SJ 44324361 Ki = 2.7 nM T60693 CT39YA 44324362 Ki = 2.4 nM T60693 CR8K3D 44326480 Ki = 0.29 nM T60693 C5NHT1 44329096 Ki = 300 nM T60693 CV57DK 44329162 Ki = 38 nM T60693 C8ABT2 44329206 Ki > 14000 nM T60693 CH46CQ 44329417 Ki = 4500 nM T60693 CV91DR 44329508 Ki > 10000 nM T60693 CL3B0J 44329509 Ki = 1000 nM T60693 C1LOP6 44329524 Ki = 3200 nM T60693 C2JOC8 44329698 Ki = 580 nM T60693 CV90JY 44329722 Ki = 3800 nM T60693 C9YU3Z 44329726 Ki > 7000 nM T60693 COE92S 44329727 Ki > 7000 nM T60693 COR3H8 44329728 Ki = 3100 nM T60693 CWD3C4 44331290 EC50 = 141 nM T60693 CHQ83J 44331291 EC50 > 10000 nM T60693 CL93FN 44331333 EC50 > 10000 nM T60693 C2FKH0 44331336 EC50 > 10000 nM T60693 C8GYX5 44331337 EC50 = 32 nM T60693 C8YV3N 44331349 EC50 > 10000 nM T60693 C5UA1P 44331366 EC50 = 22 nM T60693 C69FNR 44331395 EC50 = 300 nM T60693 C7K1YA 44331429 EC50 > 10000 nM T60693 CH0GS4 44331465 EC50 > 10000 nM T60693 CAS38O 44332117 Ki = 137 nM T60693 CR0UZ9 44333058 Ki = 0.19 nM T60693 CQ91FE 44334421 Ki = 8695 nM T60693 C26IAM 44336365 Ki = 0.1 nM T60693 CJ4WL1 44336602 Ki = 43.4 nM T60693 CGZ9N2 44336905 Ki = 997 nM T60693 CDJ9C5 44336988 IC50 = 68 nM T60693 CYMH75 44337108 Ki = 6037 nM T60693 CJ0I6Q 44337123 Ki = 3533 nM T60693 CPOX86 44337129 Ki = 2772 nM T60693 CT78UG 44337131 Ki = 641 nM T60693 CKGS32 44337160 IC50 > 1000 nM T60693 CO8Y5G 44337163 Ki = 3684 nM T60693 CWJC16 44337164 IC50 = 25.5 nM T60693 CBJ01F 44337212 Ki = 4219 nM T60693 C8IJM5 44337229 Ki = 2134 nM T60693 C97YKG 44337230 Ki = 4099 nM T60693 C3B4WO 44337231 Ki = 1841 nM T60693 CU8IY3 44337232 Ki = 1484 nM T60693 C3GQ1S 44337243 IC50 = 274 nM T60693 C3M0QX 44337249 Ki = 4125 nM T60693 C0MJL2 44337252 Ki = 4262 nM T60693 CVE93R 44337264 IC50 > 1000 nM T60693 CL27XI 44337269 IC50 = 27.2 nM T60693 CVS69U 44337271 IC50 = 116 nM T60693 C14LMK 44337273 IC50 = 184 nM T60693 CM5YJ1 44337274 IC50 = 162 nM T60693 C0XI3O 44337275 IC50 = 126 nM T60693 C5D6QW 44337276 IC50 = 10.8 nM T60693 CB1U3P 44337314 IC50 = 5.01 nM T60693 CPHU86 44337316 IC50 = 171 nM T60693 CU35AM 44337344 IC50 = 4.5 nM T60693 CB85KA 44337351 Ki = 7718 nM T60693 CI13YG 44337357 Ki = 607 nM T60693 CW2FZ7 44337362 Ki = 1341 nM T60693 CJ08FM 44337379 Ki = 3432 nM T60693 CIP87K 44337437 Ki = 2855 nM T60693 CR62KO 44337452 Ki = 7172 nM T60693 C9CIP3 44337459 Ki = 3251 nM T60693 CFA2Q7 44337460 Ki = 2240 nM T60693 CF96JK 44337473 Ki = 2938 nM T60693 CX87AS 44337513 Ki = 3911 nM T60693 CP1VN3 44337550 Ki = 1945 nM T60693 CZ02BO 44337551 Ki = 2993 nM T60693 C4AIE7 44337613 Ki = 0.2 nM T60693 CHB64V 44337616 Ki = 8.13 nM T60693 C35PQC 44337617 Ki = 6.33 nM T60693 CKZ03N 44337618 Ki = 12.32 nM T60693 C7A9FQ 44337642 Ki = 440 nM T60693 C6AVW4 44337643 Ki = 2.11 nM T60693 C8OFG5 44337644 Ki = 6.18 nM T60693 C59RIN 44337645 Ki = 28.4 nM T60693 C18MWY 44337673 Ki = 1.57 nM T60693 CI8AT5 44337683 Ki = 0.14 nM T60693 C0J9UR 44337749 Ki = 10.33 nM T60693 CJTU61 44337750 Ki = 21.89 nM T60693 CMGC86 44337764 Ki = 0.28 nM T60693 CI48SV 44337765 Ki = 0.68 nM T60693 CVP73N 44337783 Ki = 1.6 nM T60693 C7Q4HS 44337789 Ki = 34.6 nM T60693 CP4A0K 44337800 Ki = 0.61 nM T60693 C64JKH 44337822 Ki = 5.61 nM T60693 C20HGO 44337823 Ki = 1.44 nM T60693 C40VWE 44337830 Ki = 0.25 nM T60693 C3QGP4 44337831 Ki = 1.39 nM T60693 CHVG85 44337832 Ki = 2.21 nM T60693 CS57JZ 44337839 Ki = 239 nM T60693 C9CIL3 44339409 EC50 > 10000 nM T60693 CW56BK 44339424 Ki = 4153 nM T60693 C4POK5 44339425 Ki = 6000 nM T60693 CF1HE6 44339472 EC50 > 10000 nM T60693 CFRJ92 44339475 EC50 = 4.51 nM T60693 C68ZSO 44339521 EC50 > 10000 nM T60693 CX93QM 44339562 Ki > 10000 nM T60693 CO9IF8 44339563 Ki > 10000 nM T60693 C7E4MS 44339576 Ki = 1653 nM T60693 C2PDT6 44339596 Ki = 4240 nM T60693 CM42BN 44341722 Ki = 12.29 nM T60693 CND5T9 44341920 Ki = 21.08 nM T60693 CM4NE8 44342057 IC50 = 32 nM T60693 C6BX2A 44342141 IC50 = 1060 nM T60693 CD9ZS8 44342270 IC50 = 270 nM T60693 C4N6GE 44342597 Ki = 709 nM T60693 C0Z9DY 44342598 Ki = 77 nM T60693 CSZ34A 44342661 Ki = 32 nM T60693 CJVN97 44342684 Ki = 2265 nM T60693 CP97HW 44342724 Ki = 723 nM T60693 C2EQZ1 44342741 Ki = 738 nM T60693 CYTQ61 44342743 Ki = 2265 nM T60693 C0IJN7 44342746 Ki = 2265 nM T60693 CQ5B8R 44342747 Ki = 2265 nM T60693 CW5RB3 44342753 Ki = 3776 nM T60693 C1LQR9 44342754 Ki = 3776 nM T60693 CD3F2N 44342792 Ki = 783 nM T60693 CC1X5F 44342793 Ki = 452 nM T60693 C46PTB 44342843 Ki = 2265 nM T60693 CNO76C 44342910 Ki = 17 nM T60693 C5NQP9 44342911 Ki = 2 nM T60693 CNG79I 44342912 Ki = 23 nM T60693 CLC0Z1 44342925 Ki = 43 nM T60693 C74GDW 44342933 Ki = 4.9 nM T60693 CG1X6K 44342934 Ki = 16 nM T60693 CYKC24 44348604 IC50 = 336 nM T60693 CUH0O6 44348653 IC50 = 362 nM T60693 C5V9HZ 44348654 IC50 > 10000 nM T60693 CH20CJ 44348661 IC50 = 804 nM T60693 C4QNF1 44348680 IC50 > 10000 nM T60693 C0R9AD 44348681 IC50 = 6477 nM T60693 C1XQK2 44348688 IC50 > 10000 nM T60693 CE23CP 44348690 IC50 = 5436 nM T60693 C7HUL9 44348729 IC50 = 359 nM T60693 CH2FW7 44348730 IC50 = 1767 nM T60693 CY2LE5 44348770 IC50 = 2309 nM T60693 CZFN96 44348778 IC50 = 1747 nM T60693 C18CFL 44348779 IC50 = 341 nM T60693 CJM72K 44348780 IC50 = 276 nM T60693 CIO4J1 44348783 IC50 = 4424 nM T60693 C3WR5N 44348784 IC50 = 3744 nM T60693 C2GRT1 44348793 IC50 = 1941 nM T60693 C0JWA6 44348797 IC50 = 85 nM T60693 CT1OH9 44348802 IC50 = 3456 nM T60693 CA4K6J 44348815 IC50 = 2479 nM T60693 C3SF7B 44348818 IC50 = 1140 nM T60693 C91JOC 44348819 IC50 = 999 nM T60693 C0HUF9 44348820 IC50 = 827 nM T60693 C42NMT 44348821 IC50 = 738 nM T60693 CO2G7P 44348827 IC50 = 3641 nM T60693 CW8UX5 44348828 IC50 = 219 nM T60693 CRK47E 44348839 IC50 = 185 nM T60693 CZ29AH 44348841 IC50 = 5026 nM T60693 CKA9N0 44348842 IC50 = 3872 nM T60693 C7AQW3 44348843 IC50 = 924 nM T60693 CG6VS1 44348853 IC50 = 1568 nM T60693 CV29OE 44348855 IC50 = 238 nM T60693 CLE46S 44348856 IC50 = 4923 nM T60693 C6O1WU 44348862 IC50 = 1523 nM T60693 CMG0Z7 44348863 IC50 = 1492 nM T60693 C1TXV8 44348864 IC50 = 1206 nM T60693 CD9R6W 44348868 IC50 = 524 nM T60693 C9LWP3 44348876 IC50 = 560 nM T60693 CL9CI0 44348877 IC50 = 502 nM T60693 CUZL08 44348885 IC50 = 547 nM T60693 C7SAT4 44348889 IC50 = 425 nM T60693 C7EVC9 44348891 IC50 = 369 nM T60693 CTP06H 44348899 IC50 = 365 nM T60693 CRA40V 44348956 IC50 = 5061 nM T60693 CF6SQ8 44348967 IC50 = 4482 nM T60693 C1FI2W 44349005 IC50 > 10000 nM T60693 CPV8R3 44349947 Ki = 0.37 nM T60693 CX8OV0 44358749 Ki = 1100 nM T60693 C9QT7R 44358763 Ki = 1300 nM T60693 CZRQ16 44358764 Ki = 1400 nM T60693 CT6IW3 44358829 Ki = 220 nM T60693 CR7B2P 44358857 Ki = 460 nM T60693 C1UXN9 44358875 Ki = 100 nM T60693 C84JQO 44358880 Ki = 5.4 nM T60693 CYK75T 44358889 Ki = 120 nM T60693 CD2KB4 44358890 Ki = 140 nM T60693 CG7H8O 44358892 Ki = 120 nM T60693 C5R1NH 44358904 Ki = 190 nM T60693 CI0Q7R 44358923 Ki = 210 nM T60693 C1JUA9 44358924 Ki = 600 nM T60693 CYK1G5 44358967 Ki = 300 nM T60693 C0X9FD 44358968 Ki = 140 nM T60693 CG68ZO 44358969 Ki = 840 nM T60693 CHY6F1 44359130 Ki = 140 nM T60693 C8H1FC 44359131 Ki = 210 nM T60693 CX36MB 44364216 IC50 = 1400 nM T60693 CFZ95L 44364261 IC50 > 10000 nM T60693 CO2PC3 44364275 IC50 = 300 nM T60693 CF6NI2 44364277 IC50 = 160 nM T60693 CI7RP1 44364278 IC50 = 390 nM T60693 C1V4DS 44364294 IC50 = 110 nM T60693 CLV3B7 44364394 IC50 = 1.7 nM T60693 C3ZS6Q 44366280 Ki = 75 nM T60693 C1C3WO 44366432 Ki = 1.2 nM T60693 CU8MZ9 44366433 Ki = 467 nM T60693 CD18TR 44366689 Ki = 1085 nM T60693 CYL95J 44366690 Ki = 441 nM T60693 C7IFR8 44366822 Ki = 78 nM T60693 CL1JV2 44366823 Ki = 190 nM T60693 COEC43 44367007 Ki > 10000 nM T60693 CTY04M 44367017 Ki = 45 nM T60693 CT71JB 44367028 Ki = 108 nM T60693 C30QSI 44367136 Ki = 120 nM T60693 C8IZ2L 44367182 Ki = 187 nM T60693 CRO21Y 44367308 Ki = 191 nM T60693 C8BX2S 44367339 Ki = 183 nM T60693 CF5Q6M 44368739 Ki = 0.19 nM T60693 C7EMY8 44368740 Ki = 6.6 nM T60693 C7XG9B 44380504 Ki = 2.4 nM T60693 CL89XO 44380683 Ki = 160 nM T60693 CCX1K8 44380752 Ki = 940 nM T60693 CE0C5H 44380980 EC50 = 3.3 nM T60693 CT84GR 44380994 EC50 = 5.9 nM T60693 CV6E7J 44381061 Ki > 10000 nM T60693 CB26OS 44381112 EC50 = 10 nM T60693 CK8SV3 44381244 Ki = 7 nM T60693 C9XWY7 44387572 Ki = 140 nM T60693 CXS06T 44387573 Ki = 210 nM T60693 C51KZJ 44387581 Ki = 18 nM T60693 C6E0KR 44388804 Ki = 1.3 nM T60693 CIB1V0 44388818 Ki > 1000 nM T60693 CHRJ68 44388869 Ki > 1000 nM T60693 CP4XC8 44388870 Ki > 1000 nM T60693 CWN7L1 44388894 Ki = 43 nM T60693 C7BRH9 44388895 Ki > 1000 nM T60693 CM0R5U 44389887 Ki = 258 nM T60693 CGU06L 44389952 EC50 = 0.76 nM T60693 C7FE9Q 44389953 Ki = 99 nM T60693 CYV23M 44389957 Ki = 20 nM T60693 CIPC92 44389964 EC50 = 1.98 nM T60693 CIXS37 44389965 Ki = 48 nM T60693 CA01MB 44389966 Ki = 138 nM T60693 C0E8RJ 44389971 Ki = 84 nM T60693 C6JP9H 44389972 Ki = 16.3 nM T60693 CKYB47 44389976 Ki = 856 nM T60693 C95QYK 44389981 EC50 = 3.85 nM T60693 C6TF3Z 44389984 EC50 = 2.25 nM T60693 CV9FW7 44389985 Ki = 150 nM T60693 C8L1VO 44389988 EC50 = 4.37 nM T60693 CCB63E 44389992 Ki = 178 nM T60693 CVP93A 44392551 Ki = 2.9 nM T60693 CKB57F 44392581 Ki = 0.31 nM T60693 CT01GV 44392623 Ki = 0.63 nM T60693 CY5FU7 44392625 Ki = 0.48 nM T60693 CEZS26 44392630 Ki = 9.5 nM T60693 CM08ZR 44392637 Ki = 2300 nM T60693 C5ZFX2 44394283 Ki > 2000 nM T60693 COB70L 44394284 Ki > 2000 nM T60693 C5BTZ1 44394320 Ki > 2000 nM T60693 C6DB4X 44394324 Ki > 2000 nM T60693 C2OV9B 44394344 Ki > 2000 nM T60693 C1Y3NV 44394345 Ki > 2000 nM T60693 CCR2U1 44394375 Ki > 2000 nM T60693 CQ2O6J 44394381 Ki > 2000 nM T60693 CTJ2I9 44394405 Ki > 2000 nM T60693 CLFU54 44394419 Ki > 2000 nM T60693 C0A1OW 44394487 Ki > 2000 nM T60693 C61AXY 44394529 Ki > 2000 nM T60693 CRCV49 44394559 Ki > 2000 nM T60693 CJ67BT 44395278 Ki = 35 nM T60693 C3ZU0J 44395300 Ki = 17 nM T60693 CF3Z6S 44395322 Ki = 800 nM T60693 CTX47M 44395348 Ki = 0.2 nM T60693 C7T9EV 44395396 Ki = 12 nM T60693 CL6WV3 44398138 Ki = 650 nM T60693 CJ98TY 44398175 Ki = 1930 nM T60693 CRL7Y5 44399273 Ki = 57 nM T60693 C56JOK 44399274 EC50 = 1.3 nM T60693 C3M4XI 44399378 Ki = 10 nM T60693 CPSF28 44399379 Ki = 8.7 nM T60693 C1NX9P 44399492 EC50 = 19 nM T60693 CC1UY9 44399493 Ki = 1.3 nM T60693 C4XEQ2 44399584 Ki = 12 nM T60693 CR0G7H 44399648 Ki = 2.8 nM T60693 CT2YO6 44399674 Ki = 10 nM T60693 CMA91N 44399675 Ki = 1.9 nM T60693 C9GF1J 44399730 Ki = 6.1 nM T60693 CXR91I 44401402 Ki = 23 nM T60693 CQRZ78 44401457 Ki = 0.27 nM T60693 C3Y4MD 44401653 Ki = 2.2 nM T60693 C1B4QL 44403095 Ki > 10000 nM T60693 C1YL7Z 44403098 Ki > 10000 nM T60693 CFV98A 44403101 Ki > 10000 nM T60693 C6OY9S 44403102 Ki > 10000 nM T60693 CH4SX6 44403105 Ki > 10000 nM T60693 C12FIH 44403106 Ki > 10000 nM T60693 CJI6H5 44403363 Ki > 1000 nM T60693 C1URK2 44403371 Ki > 1000 nM T60693 C4DF2U 44403372 Ki > 1000 nM T60693 C26AMS 44403380 Ki > 1000 nM T60693 CL0YC4 44403381 Ki > 1000 nM T60693 C8MR3I 44403387 Ki = 48.6 nM T60693 C0XMN1 44403388 Ki = 28.5 nM T60693 CNC5T3 44403444 Ki = 475 nM T60693 CE6BH5 44403453 Ki > 1000 nM T60693 CJ61HL 44403457 Ki > 1000 nM T60693 C92NXK 44403458 Ki = 26.9 nM T60693 C4IO8C 44403459 Ki > 1000 nM T60693 C8EI5J 44403460 EC50 = 227 nM T60693 CUP2N3 44403461 Ki > 1000 nM T60693 C1YV4T 44403463 Ki > 1000 nM T60693 C8XQ5S 44403464 Ki = 210 nM T60693 C8CGE9 44403465 Ki > 1000 nM T60693 CCX98K 44403466 Ki > 1000 nM T60693 CY67AT 44403497 Ki > 1000 nM T60693 CU6EK2 44403503 Ki > 1000 nM T60693 C5XCY0 44403504 Ki = 201 nM T60693 CB15ST 44403509 Ki > 1000 nM T60693 CUW0A7 44403510 Ki > 1000 nM T60693 CS1OT5 44403515 Ki > 1000 nM T60693 COMZ82 44403520 EC50 = 58.2 nM T60693 C5NUF4 44403521 Ki = 110 nM T60693 CKS08A 44403526 Ki > 1000 nM T60693 CTUN13 44403531 Ki > 1000 nM T60693 C2U5YH 44403537 Ki > 1000 nM T60693 C4PH7R 44403545 Ki > 1000 nM T60693 CJ5S8G 44403546 Ki > 1000 nM T60693 C4LKC1 44404394 Ki > 10000 nM T60693 C3EJ4G 44404396 Ki > 10000 nM T60693 CILB28 44404652 IC50 = 430 nM T60693 CA58SU 44404670 IC50 = 1100 nM T60693 C83PCH 44404679 IC50 = 640 nM T60693 CU0YX9 44404684 IC50 = 1220 nM T60693 CEJ7F8 44404689 IC50 = 120 nM T60693 CODG94 44404695 IC50 = 2380 nM T60693 CD79WM 44404698 IC50 = 540 nM T60693 C0BED6 44404699 IC50 = 560 nM T60693 C2NHS0 44404707 IC50 = 4000 nM T60693 CNX5T8 44404731 IC50 = 2640 nM T60693 CE41AD 44405138 Ki = 1.7 nM T60693 CN0G4K 44405139 Ki = 1.6 nM T60693 CE81GQ 44405140 Ki = 490 nM T60693 CU02RP 44405141 Ki = 52.4 nM T60693 CUIG59 44405142 Ki = 130 nM T60693 CA2B3X 44405144 Ki = 30.5 nM T60693 C1UZE3 44405145 Ki = 17 nM T60693 CYX81F 44405161 Ki = 18.8 nM T60693 C14OGA 44405162 Ki = 1.6 nM T60693 CHU8N9 44405164 Ki = 14.2 nM T60693 C0AXJ5 44405165 Ki = 24.5 nM T60693 CV5Y3I 44405172 Ki = 31 nM T60693 C32CVQ 44405173 Ki = 3.3 nM T60693 CE43NQ 44405175 Ki = 5.8 nM T60693 CM05NC 44406109 Ki = 242 nM T60693 CA0RM2 44406110 Ki = 858 nM T60693 C2T6WY 44406111 Ki = 318 nM T60693 C5P9NO 44406128 Ki = 1877 nM T60693 CI2C5K 44406161 Ki = 1185 nM T60693 CRL3P8 44406171 Ki > 4652 nM T60693 CQ2D6B 44406177 Ki = 148 nM T60693 CALG92 44406185 Ki = 2156 nM T60693 C7WQ5V 44406186 Ki = 2059 nM T60693 CBH5G9 44406215 Ki = 46 nM T60693 CRI8L5 44406219 Ki > 465 nM T60693 CUH65A 44406224 Ki = 782 nM T60693 CF61YM 44406225 Ki = 152 nM T60693 CKS9V8 44406273 Ki = 116 nM T60693 CS7KQ8 44406280 Ki > 4652 nM T60693 CLE5R9 44406285 Ki = 397 nM T60693 CZFM30 44406286 Ki = 334 nM T60693 C0C2BN 44406353 Ki = 40 nM T60693 CJ6H4U 44406370 Ki = 2012 nM T60693 C79UVP 44406376 Ki > 4652 nM T60693 C4RJY2 44406656 Ki = 130 nM T60693 CSMQ84 44406657 Ki = 1.2 nM T60693 CSF2Y6 44406658 Ki = 0.38 nM T60693 C2KBP7 44406663 Ki = 0.15 nM T60693 C3SEN7 44406695 Ki = 0.62 nM T60693 C2MR7W 44406696 Ki = 0.29 nM T60693 C4LA2U 44406703 Ki = 1.2 nM T60693 COG8U3 44406710 Ki = 3.8 nM T60693 CZC51G 44406712 Ki = 7.5 nM T60693 CPO9T5 44406713 Ki = 7.3 nM T60693 CRE4Q9 44406723 Ki = 0.11 nM T60693 C4N1MC 44406724 Ki = 0.3 nM T60693 CB30EK 44406732 Ki = 0.23 nM T60693 CVER25 44407299 Ki = 710 nM T60693 C9AU3C 44407301 Ki = 110 nM T60693 CVP98E 44407305 Ki = 290 nM T60693 C4J3VF 44407309 Ki = 920 nM T60693 C3NG6O 44407310 Ki = 790 nM T60693 C7YM3D 44407311 Ki = 74 nM T60693 C2QNC5 44407312 Ki = 220 nM T60693 C3DQ8W 44407313 Ki = 270 nM T60693 CQ9X8L 44407315 Ki = 100 nM T60693 CX82DC 44407316 Ki = 260 nM T60693 CD9R7C 44407317 Ki = 690 nM T60693 CY3EH0 44407318 Ki = 360 nM T60693 CU6D4P 44407323 Ki > 1000 nM T60693 CJ51HQ 44407324 Ki = 200 nM T60693 C2I8RZ 44407329 Ki = 510 nM T60693 CW89MA 44407330 Ki = 620 nM T60693 CTLY61 44407348 Ki = 200 nM T60693 CE9K1V 44407351 Ki > 1000 nM T60693 CY8R2X 44407359 Ki = 360 nM T60693 C69OZA 44407360 Ki = 610 nM T60693 CB16YW 44407361 Ki = 570 nM T60693 C2P4ZH 44407364 Ki = 150 nM T60693 C59XVU 44411613 Ki = 840 nM T60693 CYE4D3 44411762 Ki = 410 nM T60693 CMG79P 44411790 Ki = 8530 nM T60693 CS0ZC2 44411794 Ki = 56 nM T60693 CDK08M 44411860 Ki = 1620 nM T60693 C52WZH 44413231 Ki > 10000 nM T60693 CFJ64A 44413232 Ki = 1900 nM T60693 CNFC81 44413248 Ki > 5000 nM T60693 C0V4FI 44413286 Ki = 3890 nM T60693 CS7BI8 44413301 Ki > 5000 nM T60693 C1NGS0 44413314 Ki > 5000 nM T60693 C5J0BU 44413315 Ki > 5000 nM T60693 CH7E1C 44413329 Ki > 5000 nM T60693 C1OQ0L 44413330 Ki = 4300 nM T60693 CKV5S0 44413361 Ki > 5000 nM T60693 C5PHK7 44413362 Ki > 5000 nM T60693 CSQZ28 44413379 Ki = 1010 nM T60693 CCU2B5 44413384 Ki = 1170 nM T60693 CD5SZ9 44413385 Ki = 2600 nM T60693 C7GE2K 44413395 Ki > 5000 nM T60693 CCK6Y5 44413396 Ki > 5000 nM T60693 C0FL8K 44413401 Ki > 5000 nM T60693 C6J3HP 44413402 Ki > 5000 nM T60693 CB2OJ9 44413408 Ki > 5000 nM T60693 C82VJB 44413413 Ki > 5000 nM T60693 CP31JV 44413414 Ki = 710 nM T60693 C98OQG 44413423 Ki = 750 nM T60693 CH0DS7 44413441 Ki = 330 nM T60693 CLSK72 44413442 Ki = 680 nM T60693 CL4YP0 44413961 EC50 = 1.84 nM T60693 C3W9ZR 44415103 IC50 = 1048 nM T60693 C5XA2V 44415104 IC50 = 10516 nM T60693 C5DQU3 44415132 IC50 = 2358 nM T60693 CHA92Z 44415133 IC50 = 14430 nM T60693 CW97YG 44415143 IC50 = 11130 nM T60693 CPL8U5 44415144 IC50 = 10635 nM T60693 CXAN82 44415167 IC50 = 32160 nM T60693 CSW4K9 44415190 IC50 = 1450 nM T60693 C7JI0K 44415191 IC50 = 9674 nM T60693 C1DH7S 44415192 IC50 = 22559 nM T60693 CNW4V0 44415202 IC50 = 22457 nM T60693 C3UC4M 44415224 IC50 = 3855 nM T60693 CNT96C 44415298 IC50 = 22435 nM T60693 C7EHS3 44415299 IC50 = 15589 nM T60693 C5Y7KT 44415300 IC50 = 4141 nM T60693 CCX92L 44415312 IC50 = 6059 nM T60693 CU65WM 44415621 Ki = 27 nM T60693 C1MO6K 44415676 Ki = 8.5 nM T60693 C7U8LB 44415720 Ki = 36 nM T60693 CGZ0A6 44415722 Ki > 10000 nM T60693 CT1U6D 44415744 Ki > 10000 nM T60693 CB7OZ0 44415762 Ki = 641 nM T60693 CY04UN 44415763 Ki = 665 nM T60693 C1UT9Q 44415832 Ki = 1.3 nM T60693 C2Z9JF 44415854 Ki = 6.9 nM T60693 CDC04T 44415855 Ki = 240 nM T60693 C35XWU 44415862 Ki > 10000 nM T60693 CEW6B0 44415863 Ki > 10000 nM T60693 CEB17O 44415873 Ki = 328 nM T60693 C59QWV 44415874 Ki = 65.2 nM T60693 C9EJK4 44415878 Ki = 1000 nM T60693 C58VYH 44415884 Ki > 10000 nM T60693 CXI3Y8 44415888 Ki = 17.6 nM T60693 CM5E2V 44415889 Ki = 168 nM T60693 COA76L 44415897 Ki > 10000 nM T60693 C1RHI9 44415907 Ki > 10000 nM T60693 CF8VL9 44415908 Ki = 223 nM T60693 CF48RT 44415931 Ki > 10000 nM T60693 CF8G6R 44415932 Ki = 28.9 nM T60693 CK26WT 44415935 Ki > 10000 nM T60693 C8LUO6 44415936 Ki > 10000 nM T60693 C5M4JI 44415946 Ki = 2.3 nM T60693 CBU7I8 44415950 Ki > 10000 nM T60693 C9E5KT 44415951 Ki = 769 nM T60693 CLB03N 44415968 Ki > 10000 nM T60693 CN3MW0 44415987 Ki > 10000 nM T60693 CF3B9X 44416009 Ki = 376 nM T60693 CIKJ32 44416013 Ki = 374 nM T60693 CG5VA4 44416030 EC50 = 2.4 nM T60693 C8K2SQ 44416049 Ki > 1000 nM T60693 C6CRQ4 44416051 EC50 = 25.2 nM T60693 C5LUE3 44416052 EC50 = 37.2 nM T60693 C31EBI 44416118 Ki = 220 nM T60693 C0P3OR 44416128 Ki = 90.9 nM T60693 COT14P 44416129 Ki = 332 nM T60693 CB7QZ6 44416134 Ki > 10000 nM T60693 CVPL90 44416144 Ki = 117 nM T60693 C6V9RO 44416145 Ki = 16.5 nM T60693 CNX96O 44416154 Ki = 1392 nM T60693 CUF36X 44417374 Ki = 0.91 nM T60693 CFJC63 44417384 Ki = 53.6 nM T60693 C7AMJ6 44419172 Ki > 1000 nM T60693 C6TWB4 44419173 Ki > 1000 nM T60693 CX3W7M 44419181 Ki > 1000 nM T60693 C4RZ8O 44419189 Ki > 1000 nM T60693 CM2P1G 44419196 Ki > 1000 nM T60693 CVW98H 44419201 Ki > 1000 nM T60693 C51WAF 44419209 Ki > 1000 nM T60693 C09YMI 44419228 Ki > 1000 nM T60693 CG3E9L 44419233 Ki > 1000 nM T60693 CB3O2R 44419236 Ki > 1000 nM T60693 C9JL8N 44419242 Ki = 221 nM T60693 CK9VL4 44419243 Ki > 1000 nM T60693 CP2E7J 44419244 Ki > 1000 nM T60693 CVS42X 44419245 Ki > 1000 nM T60693 C8LP4T 44419248 EC50 = 210 nM T60693 C6MIS5 44419256 Ki > 1000 nM T60693 CB9J0U 44419257 Ki > 1000 nM T60693 C8AI5Q 44419258 Ki > 1000 nM T60693 CYP8J7 44419289 Ki > 1000 nM T60693 CKD2A9 44419291 Ki > 1000 nM T60693 CG9W6L 44419292 Ki > 1000 nM T60693 C72HIJ 44421393 Ki = 18.5 nM T60693 C0M1LF 44421396 Ki = 24.3 nM T60693 CI12ZC 44421399 Ki = 7.38 nM T60693 COM3F5 44421400 Ki = 2.51 nM T60693 C2L4MW 44421401 Ki = 6.29 nM T60693 CKA1J2 44421403 Ki = 24.9 nM T60693 C5S4EC 44421406 Ki = 8.97 nM T60693 CW6I0V 44421407 Ki = 89.1 nM T60693 CN6E4Q 44421408 EC50 = 98.2 nM T60693 CLEH29 44421409 Ki = 289 nM T60693 C4ZXO2 44421412 EC50 = 153 nM T60693 C5K6YB 44421422 EC50 = 131 nM T60693 C9ACE6 44422807 Ki = 0.34 nM T60693 C2IE1L 44422808 Ki = 0.12 nM T60693 C0Q8TZ 44425152 Ki > 10000 nM T60693 C4NWJ9 44425154 Ki > 10000 nM T60693 CYQ28K 44425156 Ki = 990 nM T60693 CV7N0H 44425963 Ki = 6.5 nM T60693 C10OMS 44426811 Ki = 185 nM T60693 C49KAS 44426813 Ki = 312 nM T60693 CJ5FC0 44426816 Ki = 1771 nM T60693 C4TFP1 44426818 Ki = 6753 nM T60693 CP5V8D 44426821 Ki = 4381 nM T60693 C5L4SE 44426822 Ki = 5935 nM T60693 C36SCP 44426823 Ki = 2993 nM T60693 C72RXV 44426824 Ki = 971 nM T60693 C0S5TE 44426829 Ki = 1362 nM T60693 CL1EG2 44426830 Ki = 6621 nM T60693 CBFY73 44426831 Ki = 4294 nM T60693 CFO9Q6 44426832 Ki = 535 nM T60693 C2NFA4 44426833 Ki = 1971 nM T60693 COJ48Z 44426834 Ki = 164 nM T60693 CUD42S 44426835 Ki = 1479 nM T60693 CKJ90O 44426836 Ki = 1144 nM T60693 CZ4R6J 44426837 Ki = 2443 nM T60693 CPDE73 44426838 Ki = 1174 nM T60693 C53JGK 44426839 Ki = 8057 nM T60693 C7IJY0 44426840 Ki = 1172 nM T60693 CJB90W 44426841 Ki = 123 nM T60693 CK3B6E 44426843 Ki = 306 nM T60693 CD3TB8 44426844 Ki = 2878 nM T60693 CFY3A6 44427433 Ki = 18 nM T60693 C0M4EP 44427434 Ki = 0.65 nM T60693 CT2Z8J 44429058 Ki = 52 nM T60693 CQ87UY 44429059 Ki = 6.6 nM T60693 CF5OJ0 44430021 Ki = 61045 nM T60693 CUQ95Y 44430022 Ki = 2769 nM T60693 CZA0E6 44430023 Ki = 1658 nM T60693 CWX67P 44430033 Ki = 2574 nM T60693 C40BHT 44430038 Ki = 15 nM T60693 C1QXR6 44430040 Ki = 725 nM T60693 CS6Y5Z 44430042 Ki = 425 nM T60693 C4CHV5 44430043 Ki = 279 nM T60693 CX9P5R 44430044 Ki = 450 nM T60693 CA51JN 44430045 Ki = 1056 nM T60693 C2G9HQ 44430046 Ki = 2092 nM T60693 C8PI4A 44430047 Ki = 771 nM T60693 CL1N4D 44430048 Ki = 664 nM T60693 C0AYM6 44430049 Ki = 1354 nM T60693 CMJT74 44430050 Ki = 255 nM T60693 C4ZG6A 44430079 Ki = 215 nM T60693 CSNQ43 44430080 Ki = 330 nM T60693 CXV9J7 44430081 Ki = 323 nM T60693 CFHY18 44430083 Ki = 261 nM T60693 C6SBE1 44430084 Ki = 139 nM T60693 CXZ2D3 44430085 Ki = 146 nM T60693 CI4X3Z 44430087 Ki = 186 nM T60693 C15KTO 44432560 Ki = 1008 nM T60693 C9KQE6 44432562 Ki = 621 nM T60693 CJN2O9 44432597 Ki = 188 nM T60693 CM3P1O 44432599 Ki = 121 nM T60693 C37YLC 44432606 Ki = 84 nM T60693 CA9S4M 44432608 Ki = 121 nM T60693 CG7KL2 44432609 Ki = 366 nM T60693 CLQH28 44432610 Ki = 201 nM T60693 C3W6AY 44432611 Ki > 4652 nM T60693 CC15LP 44432614 Ki = 3116 nM T60693 C34OTB 44433399 Ki = 64 nM T60693 CT4QL9 44433400 Ki = 26 nM T60693 CO08LU 44433401 Ki = 170 nM T60693 CC5G2Y 44433402 Ki = 230 nM T60693 CJ20NZ 44434062 Ki = 2150 nM T60693 CF78VR 44434063 Ki = 1221 nM T60693 C38NOM 44434064 Ki = 555.9 nM T60693 CT8QH4 44434065 Ki = 2428.17 nM T60693 CTM38X 44434066 Ki = 3606 nM T60693 CMT4U1 44434067 Ki = 360.6 nM T60693 CF0V8Z 44434068 Ki = 2873 nM T60693 C3H1NC 44434069 Ki > 4897 nM T60693 C38LOE 44434072 Ki = 105.88 nM T60693 CR9GY1 44434075 Ki = 116.41 nM T60693 CT6ZD0 44434077 Ki = 78.09 nM T60693 COI7A6 44434079 Ki = 105.95 nM T60693 C73FSU 44434081 Ki = 318.95 nM T60693 CKEY87 44434082 Ki = 71.62 nM T60693 CLZ68X 44434084 Ki = 61.65 nM T60693 C20PXC 44434087 Ki = 703.78 nM T60693 C1KB9R 44434088 Ki = 359.89 nM T60693 CLU1X5 44434089 Ki = 3254 nM T60693 CZM8I9 44434201 EC50 = 2700 nM T60693 CB2AQ4 44434932 Ki > 5000 nM T60693 C81KMS 44434933 Ki > 5000 nM T60693 COEG19 44434934 Ki > 5000 nM T60693 C9XW8Q 44434935 Ki > 5000 nM T60693 C4N9OY 44434936 Ki > 5000 nM T60693 C5UG8I 44434937 Ki > 5000 nM T60693 CGLY08 44434938 Ki = 1147.5 nM T60693 C92WQA 44434939 Ki > 5000 nM T60693 C04LKG 44434940 Ki > 5000 nM T60693 CT95NA 44434941 Ki = 2808.74 nM T60693 CGKC17 44434942 Ki > 5000 nM T60693 CVF9O5 44434943 Ki > 5000 nM T60693 CUA32P 44434944 Ki = 23.34 nM T60693 CRBX46 44434945 Ki = 24.15 nM T60693 CD0R6I 44434947 Ki > 1000 nM T60693 CIN4E6 44434948 Ki > 1000 nM T60693 CZB4Q9 44438912 Ki = 517 nM T60693 C7RD2E 44438916 Ki = 26.2 nM T60693 CNL30S 44438917 Ki = 16.4 nM T60693 C5D4NZ 44438920 Ki = 50 nM T60693 CA2LD5 44438921 Ki = 60.5 nM T60693 C6H7AD 44438922 Ki = 22.5 nM T60693 CRN3W4 44438961 Ki = 13 nM T60693 CGYD89 44438962 Ki = 25.5 nM T60693 CZ48KD 44438963 Ki = 776 nM T60693 C2EGK7 44438964 Ki = 1183 nM T60693 COX57F 44438965 Ki = 1086 nM T60693 C9S2HB 44438966 Ki = 579 nM T60693 C1HF6E 44438967 Ki = 3529 nM T60693 C3L7SB 44438968 Ki = 1602 nM T60693 CE63GK 44438971 Ki = 4628 nM T60693 C8TVI4 44438974 Ki = 858 nM T60693 CPHS56 44438975 Ki = 1448 nM T60693 CK3Z5G 44438978 Ki = 2009 nM T60693 CPA4U5 44438983 Ki = 145 nM T60693 C2TKY5 44438988 Ki = 13.7 nM T60693 CL7WN5 44438993 Ki = 143 nM T60693 C0A2OM 44439000 Ki = 282 nM T60693 CMQA60 44439001 Ki = 169 nM T60693 CH57IQ 44439874 Ki > 10000 nM T60693 CNS7T5 44439878 Ki > 10000 nM T60693 CF8K5H 44441067 Ki = 74 nM T60693 CM9I8H 44443049 Ki = 1440 nM T60693 C5CA7D 44443050 Ki > 7000 nM T60693 CF86GQ 44443051 Ki = 582 nM T60693 CHEI51 44443452 Ki = 360 nM T60693 CY78KN 44443453 Ki = 250 nM T60693 CF1IC2 44443454 Ki = 160 nM T60693 CDJ8T5 44444601 EC50 = 1.1 nM T60693 C9N8VT 44444603 Ki = 1.1 nM T60693 C57TLG 44444604 Ki = 19 nM T60693 CBR38Y 44444613 Ki = 18 nM T60693 C56QDE 44448327 EC50 = 0.11 nM T60693 CPW3J0 44448489 EC50 = 0.71 nM T60693 CN9X6W 44448522 EC50 = 0.39 nM T60693 C6TEA5 44448524 EC50 = 0.12 nM T60693 CET3O5 44448563 EC50 = 0.24 nM T60693 CT16AC 44448691 EC50 = 2000 nM T60693 C1G9ZO 44448692 EC50 = 3 nM T60693 CY8RO4 44448772 EC50 = 1000 nM T60693 C9K8EN 44448775 EC50 = 3200 nM T60693 CW7BG9 44448874 EC50 = 7900 nM T60693 CR6TO5 44448876 EC50 = 1300 nM T60693 CF40AD 44448913 EC50 = 1300 nM T60693 C5OR0Q 44448947 EC50 = 5000 nM T60693 C15VTJ 44448976 EC50 = 30000 nM T60693 C1F2MP 44449004 EC50 = 6300 nM T60693 CL9M2D 44449052 EC50 = 15000 nM T60693 CL4H8Y 44449053 EC50 = 3200 nM T60693 C3L4XD 44449079 EC50 = 5000 nM T60693 C4T1MQ 44449106 EC50 = 500 nM T60693 C9XZY1 44449107 EC50 = 7900 nM T60693 CV31WQ 44449136 EC50 = 10000 nM T60693 CA4DS0 44449171 EC50 = 1000 nM T60693 CA61WE 44449202 EC50 = 5000 nM T60693 CC19LO 44449228 EC50 = 790 nM T60693 CT39QP 44450085 IC50 = 88 nM T60693 C1SQ7M 44450086 IC50 = 31 nM T60693 CJLI69 44450262 Ki = 45.5 nM T60693 C4NFQ9 44450499 Ki = 740 nM T60693 C5W9PF 44452254 Ki = 1100 nM T60693 CVI7M0 44452281 Ki = 1700 nM T60693 CWAN90 44452282 Ki = 2400 nM T60693 CUIC24 44453700 Ki = 510 nM T60693 C6QV3U 44453726 Ki = 720 nM T60693 C5HM3F 44453728 Ki = 240 nM T60693 CDY56P 44453750 Ki = 83 nM T60693 CO56PJ 44453779 Ki = 160 nM T60693 CO2XU7 44453801 Ki = 910 nM T60693 COI2B9 44453822 Ki = 67 nM T60693 CR1S3K 44453824 Ki = 460 nM T60693 C4ID6Y 44453825 Ki = 230 nM T60693 CBUE46 44453848 Ki = 1200 nM T60693 CZ7X2D 44453849 Ki = 550 nM T60693 CTEK70 44453879 Ki = 1400 nM T60693 CH1D0B 44453880 Ki = 2200 nM T60693 CA05FK 44453881 Ki = 2200 nM T60693 CN7B2P 44453901 Ki = 690 nM T60693 C81IOK 44453925 Ki = 1100 nM T60693 C3RQ4A 44456065 Ki = 28.7 nM T60693 CP1M0U 44456146 EC50 = 10 nM T60693 CZX0U1 44456344 Ki > 1000 nM T60693 C12XGE 44456400 Ki > 10000 nM T60693 C9KU1O 44456785 Ki = 0.91 nM T60693 C6PEF7 44456833 Ki = 1.7 nM T60693 CDE47Z 44458578 IC50 = 230 nM T60693 CDYZ85 44458640 IC50 = 37 nM T60693 CW5IA3 44458656 IC50 = 49 nM T60693 C0HC1Q 44458665 IC50 = 140 nM T60693 C8YJK3 44458686 IC50 = 6.3 nM T60693 CLY6J7 44458703 IC50 = 4.6 nM T60693 C5D1CF 44458725 IC50 = 400 nM T60693 C61XFS 44458749 IC50 = 14 nM T60693 CJ84CH 44459002 IC50 = 0.22 nM T60693 C0OLA2 44459016 IC50 = 1.5 nM T60693 C3I1LF 44463491 Ki = 320 nM T60693 CQ0WM7 44469273 IC50 > 5000 nM T60693 C0N2XB 44474938 Ki = 344 nM T60693 C4L1SW 44530683 EC50 = 200 nM T60693 CL5NO6 44541248 Ki = 2.89 nM T60693 C6K3GX 44541249 EC50 = 0.3 nM T60693 CVX16Z 44541250 EC50 = 3.18 nM T60693 C29MSC 44541387 Ki = 13.7 nM T60693 CI9O3F 44541388 Ki = 2.73 nM T60693 C6TW8L 44541389 Ki = 74.4 nM T60693 C6T1UX 44551464 Ki = 0.37 nM T60693 C32AGV 44561123 EC50 = 0.2 nM T60693 CONA75 44561156 EC50 = 0.1 nM T60693 CG1W8A 44561157 EC50 = 16 nM T60693 CXH86I 44561195 EC50 = 1600 nM T60693 CD7A4H 44561196 EC50 = 320 nM T60693 C8HCR6 44561197 EC50 = 800 nM T60693 C9HG8L 44561236 EC50 = 40 nM T60693 CR5T0L 44561237 EC50 = 4000 nM T60693 CF21JK 44561238 EC50 = 100 nM T60693 CMJ60R 44561239 EC50 = 32 nM T60693 C0W4HQ 44561240 EC50 = 800 nM T60693 C6A0TH 44561276 EC50 = 160 nM T60693 C4SVU2 44561370 IC50 = 9700 nM T60693 CRJM24 44561454 IC50 > 10000 nM T60693 CXJK43 44561493 IC50 > 10000 nM T60693 CQKE48 44564372 Ki = 1012.7 nM T60693 CPH0A5 44565363 Ki = 0.34 nM T60693 CL80WF 44570025 Ki = 5.6 nM T60693 C5W8ZR 44570027 EC50 = 170 nM T60693 C8BSQ4 44570028 EC50 = 9.6 nM T60693 C9ERN6 44570030 Ki = 100 nM T60693 CP2M8D 44570031 Ki = 2.1 nM T60693 CN7UA9 44570032 Ki = 21 nM T60693 CPA48R 44570066 Ki = 19 nM T60693 C5RWA8 44570068 EC50 = 30 nM T60693 CK4JO2 44570069 EC50 = 41 nM T60693 CGK40O 44570070 Ki = 0.39 nM T60693 C6C0XR 44570071 Ki = 46 nM T60693 CT10RB 44570072 Ki = 30 nM T60693 C8P3SX 44570073 Ki = 2.1 nM T60693 CB01RQ 44570075 Ki = 100 nM T60693 C4ZCX6 44576628 IC50 = 5.3 nM T60693 C8HF3V 44577045 Ki = 580 nM T60693 CRME18 44577046 Ki = 34 nM T60693 CI1L7Y 44577047 Ki = 110 nM T60693 CDPS18 44577048 Ki = 0.7 nM T60693 C8OU4Q 44577049 Ki = 32 nM T60693 CGMC75 44577468 Ki = 1 nM T60693 CZUW31 44577469 Ki = 560 nM T60693 CES86D 44577470 Ki = 8.6 nM T60693 CU6ZT4 44577524 Ki = 240 nM T60693 CXS42P 44577525 Ki = 140 nM T60693 CWIG26 44577526 Ki = 48 nM T60693 CTIH86 44577527 Ki = 3.2 nM T60693 CXT62C 44581771 EC50 = 0.96 nM T60693 CUT4E2 44581831 EC50 = 330 nM T60693 C5DGV7 44581832 Ki = 497 nM T60693 C3M7SO 44581833 EC50 = 299 nM T60693 CRK51Y 44581834 Ki = 36 nM T60693 CV0K4M 44581870 Ki = 83 nM T60693 CT8QN6 44581871 Ki = 20 nM T60693 C2D8FN 44581872 Ki = 154 nM T60693 CN5XH2 44581873 Ki = 196 nM T60693 C7OR9A 44581900 Ki = 109 nM T60693 CG1DL2 44582176 Ki = 1012.7 nM T60693 C3YMV4 44582184 Ki = 47.81 nM T60693 CKFX03 44582185 Ki = 49.21 nM T60693 CK8G4D 44582186 Ki = 586.42 nM T60693 CIX09B 44582198 Ki > 10000 nM T60693 CC06XI 44582199 Ki = 67.15 nM T60693 CEUS82 44582200 Ki = 148.23 nM T60693 CG58FU 44582217 Ki > 1000 nM T60693 C28VHY 44582218 Ki = 46.57 nM T60693 CU6ZC7 44582249 Ki > 1000 nM T60693 CV23PR 44582250 Ki > 1000 nM T60693 CDV9E2 44582251 Ki > 1000 nM T60693 CH2SV6 44582278 Ki > 1000 nM T60693 C3K9LN 44582279 Ki > 1000 nM T60693 CM21UD 44583389 Ki = 28 nM T60693 C6YOC5 44583390 Ki = 21 nM T60693 CX1L5P 44583391 Ki = 1300 nM T60693 C7PCJ1 44583392 Ki > 1000 nM T60693 CAHK35 44583425 Ki = 270 nM T60693 C7VWA3 44583426 Ki > 1000 nM T60693 CNG34J 44583429 Ki > 1000 nM T60693 CHZ46N 44583430 Ki > 1000 nM T60693 CASI92 44583431 Ki > 1000 nM T60693 CLAR69 44583432 Ki > 1000 nM T60693 CP8HI6 44586853 EC50 = 3.2 nM T60693 CL83XM 44586854 EC50 = 1.3 nM T60693 C0YM5K 44586855 EC50 = 6.3 nM T60693 CR9MH4 44586884 EC50 = 4 nM T60693 C6KY1J 44586885 EC50 = 4000 nM T60693 CXI52S 44586886 EC50 = 7900 nM T60693 C7HQ2U 44586887 EC50 > 10000 nM T60693 CJOH07 44586888 Ki = 11 nM T60693 CJS8F2 44586890 Ki = 0.87 nM T60693 CSD27B 44586909 EC50 = 3200 nM T60693 C2E1HJ 44586910 EC50 = 630 nM T60693 C01ECK 44586911 EC50 > 10000 nM T60693 CND46S 44586912 EC50 = 250 nM T60693 CP2N8S 44586914 Ki = 0.48 nM T60693 C7P0XN 44586916 Ki = 1.3 nM T60693 CV9H6N 44586918 Ki = 0.048 nM T60693 CP8EX5 44586920 Ki = 18 nM T60693 C23PVW 44586939 EC50 = 790 nM T60693 C1BX7R 44586940 EC50 = 79 nM T60693 C9LU0Z 44586941 EC50 = 400 nM T60693 C1I0RO 44586943 Ki = 0.21 nM T60693 C5KN8O 44586945 Ki = 67 nM T60693 CZ9NA4 44586947 Ki = 8.6 nM T60693 CH97QC 44586949 Ki = 28 nM T60693 C6BMQ4 44586974 EC50 = 3 nM T60693 C9M1BS 44586975 EC50 = 1.6 nM T60693 C53UKN 44586976 EC50 = 2 nM T60693 C8NHF6 44586977 EC50 = 4 nM T60693 C8A9WK 44586979 Ki = 9 nM T60693 CZ28KA 44586981 Ki = 28 nM T60693 CYC3Z6 44586983 Ki = 5.2 nM T60693 CG2R9W 44587037 EC50 = 400 nM T60693 C9D7CL 44587038 EC50 = 1000 nM T60693 CHJ54K 44587039 EC50 = 790 nM T60693 C6BVQ9 44587040 EC50 = 630 nM T60693 CRBI42 44587179 EC50 = 2000 nM T60693 C7V5ZN 44587180 EC50 = 1000 nM T60693 CT5LJ3 44587203 EC50 = 320 nM T60693 C2W1FV 44587204 EC50 = 2000 nM T60693 C9BDZ0 44587205 EC50 = 320 nM T60693 CR8D0K 44587227 EC50 = 790 nM T60693 CGS50I 44587228 EC50 = 1300 nM T60693 CMNB42 44587259 EC50 = 2000 nM T60693 C4E9GW 44587260 EC50 = 7900 nM T60693 C1HA0F 44588005 Ki = 4820 nM T60693 CS1G0I 44588006 Ki = 200 nM T60693 CT3C8S 44588007 Ki = 560 nM T60693 CDMZ71 44588493 Ki = 10000 nM T60693 CVCW78 44588494 Ki = 78 nM T60693 CN7OR6 44588495 Ki = 910 nM T60693 CZIM85 44588496 Ki = 26 nM T60693 C6L7IF 44588748 Ki = 0.195 nM T60693 C6EQ3R 44590514 IC50 = 2209 nM T60693 CEXW79 44590551 IC50 = 707 nM T60693 C5UIT4 44590552 IC50 > 10000 nM T60693 CP83ZW 44590553 IC50 > 10000 nM T60693 C1AP0B 44590554 IC50 > 10000 nM T60693 C4U3AE 44590580 IC50 > 10000 nM T60693 CBS8P1 44590581 IC50 > 10000 nM T60693 C41SFR 44590582 IC50 = 7993 nM T60693 CD70YK 44590629 IC50 = 7136 nM T60693 CY36KS 44590630 IC50 = 1324 nM T60693 C60XNA 44590631 IC50 = 155 nM T60693 CJ3R7Q 44590632 IC50 = 6002 nM T60693 CMH26K 44590677 IC50 = 922 nM T60693 CN8S5P 44590678 IC50 = 1005 nM T60693 CFLP28 44591164 Ki = 0.063 nM T60693 C8ZC6O 44591193 Ki = 0.05 nM T60693 CEA9O2 44591194 Ki = 12 nM T60693 CER74Z 44591195 Ki = 0.81 nM T60693 CIU9T1 44591196 Ki = 0.92 nM T60693 CO3P8X 44591197 Ki = 0.51 nM T60693 CN5ZF8 44591198 Ki = 0.23 nM T60693 CZJ16A 44591987 Ki = 0.46 nM T60693 C6A1PL 44592015 Ki = 0.34 nM T60693 CB3VG2 44592016 Ki = 7.7 nM T60693 CXL41O 44592053 EC50 = 3.9 nM T60693 C3VSJ2 44592054 Ki = 210 nM T60693 CNI1E9 44592056 Ki = 6.3 nM T60693 CUW6Q3 44592086 Ki = 0.29 nM T60693 C8DS7Q 44592087 Ki = 16 nM T60693 CU5GE1 44592088 Ki = 2.3 nM T60693 C9GRS1 44592089 Ki = 19 nM T60693 CPX7G6 44592124 Ki = 47 nM T60693 CAE64R 44593421 EC50 = 4 nM T60693 CDPU87 44596170 Ki = 0.0003 nM T60693 C2EC4H 44597424 Ki = 5870 nM T60693 CJ69LZ 44597425 Ki = 9500 nM T60693 C3ASC5 44597529 Ki = 413 nM T60693 C6XHL0 44597530 Ki = 1090 nM T60693 CAOX39 44597597 Ki = 0.62 nM T60693 C2C9LF 44597714 Ki = 0.47 nM T60693 CEOB85 44597715 Ki = 2.2 nM T60693 C1R3QC 44597828 Ki = 0.94 nM T60693 CRS74M 44597830 Ki = 4.7 nM T60693 C39PTC 44597831 Ki = 0.42 nM T60693 C14EJV 44597940 Ki = 18 nM T60693 CKT8F2 44598180 Ki = 21 nM T60693 C0TNG6 44598228 Ki = 5.8 nM T60693 CE41CY 44598229 Ki = 145 nM T60693 CHL71F 44598230 Ki = 69 nM T60693 C4HB6F 44598231 Ki = 11 nM T60693 C2BGU8 44598282 Ki = 6 nM T60693 C4NPD0 44598283 Ki = 5.9 nM T60693 CLID76 44598284 Ki = 1.3 nM T60693 CV0GR9 44599826 Ki = 0.5 nM T60693 C84NFS 44599828 Ki = 1.2 nM T60693 CI6CW8 44599979 Ki = 2.6 nM T60693 CFY8I6 44599981 Ki = 11 nM T60693 C2XQN6 44599984 Ki = 3.5 nM T60693 C0G4ON 44600135 Ki = 8.6 nM T60693 C24QEG 44600140 Ki = 10 nM T60693 CQO2U6 44600308 Ki = 7.5 nM T60693 C0BIC2 44601470 Ki = 40.3 nM T60693 C3Q0ZL 44601476 IC50 = 1120 nM T60693 CVH94R 44608034 IC50 = 2930 nM T60693 CHM9C0 44620897 IC50 > 18000 nM T60693 CH68PJ 44620907 IC50 = 937 nM T60693 C3DCT2 44626536 Ki = 12 nM T60693 CUZY73 44626538 Ki = 28 nM T60693 CG8W0U 44626542 Ki = 86 nM T60693 CY6D4O 44626643 Ki = 310 nM T60693 CB9JD0 44626647 Ki = 140 nM T60693 C25QXW 44626747 Ki = 350 nM T60693 C2NC5S 44626748 Ki = 4.9 nM T60693 C6GB5A 44626749 Ki = 37 nM T60693 CCZ89E 44626842 Ki = 40 nM T60693 CKRL83 44627034 Ki = 44 nM T60693 CBNJ20 44627035 Ki = 54 nM T60693 CVD03Q 44627135 Ki = 67 nM T60693 C8XG3W 44627136 Ki = 31 nM T60693 C8PK2F 44627248 Ki = 13 nM T60693 C81KJQ 44627363 Ki = 26 nM T60693 CLUP27 44627365 Ki = 30 nM T60693 C8NJR1 44627679 Ki = 72 nM T60693 C7CJM9 44627680 Ki = 0.79 nM T60693 CM49FS 44627786 Ki = 5.8 nM T60693 C81LTN 44627787 Ki = 0.51 nM T60693 CPTL91 44627788 Ki = 3.9 nM T60693 CZ6VP4 44627789 Ki = 16 nM T60693 CQZ0W4 44627899 Ki = 0.03 nM T60693 C6AR0U 44627902 Ki = 0.59 nM T60693 CK0T4Y 44627998 Ki = 0.6 nM T60693 C79JNE 44627999 Ki = 0.99 nM T60693 CVI57S 44628102 Ki = 1.6 nM T60693 CS8X1U 44665679 IC50 = 4 nM T60693 CR3PL6 44665680 IC50 = 120 nM T60693 CT5CK8 44665687 IC50 = 70 nM T60693 C3HXK5 45100475 IC50 = 3050 nM T60693 C4LOY2 45115589 IC50 = 60 nM T60693 C98YEZ 45256309 Ki = 1303 nM T60693 C2S8TW 45256310 Ki = 84.7 nM T60693 CU8I6T 45263517 Ki = 295 nM T60693 CY0GS5 45264200 Ki = 18 nM T60693 CVDQ53 45265789 Ki = 1205 nM T60693 C40CHQ 45269407 Ki = 28.2 nM T60693 CT1U4X 45270231 Ki = 14.7 nM T60693 C7HF9D 45271055 Ki = 6.75 nM T60693 CV53JT 45479170 IC50 > 18000 nM T60693 CIL49C 45482634 Ki = 0.12 nM T60693 CAP40I 45483185 Ki = 1747 nM T60693 CMN6O9 45483211 Ki = 4796 nM T60693 CFR5M7 45483251 Ki = 4742 nM T60693 CL7KU2 45483259 Ki = 4542 nM T60693 C8DOR2 45483260 Ki = 2928 nM T60693 CFU8K5 45483286 Ki = 6666 nM T60693 C1X8JY 45483646 Ki > 10000 nM T60693 CGOZ34 45483648 Ki = 5543 nM T60693 CI8M5T 45483656 Ki > 10000 nM T60693 CE13WZ 45483658 Ki = 4249 nM T60693 CEZJ19 45483659 Ki = 6176 nM T60693 C43JND 45483664 Ki = 576 nM T60693 C49WAV 45483668 Ki = 3556 nM T60693 CVC0G3 45483672 Ki > 10000 nM T60693 C0J4CG 45483978 Ki = 0.13 nM T60693 CFY46C 45483979 Ki = 3.4 nM T60693 C89UEA 45485826 Ki = 901 nM T60693 C76IZT 45485837 Ki = 3606 nM T60693 C2DRY1 45485876 Ki = 2549 nM T60693 CBW8D7 45485877 Ki = 6405 nM T60693 C2OE9C 45485974 Ki = 7081 nM T60693 CBP10O 45485982 Ki = 4985 nM T60693 CS2IC5 45485986 Ki > 10000 nM T60693 CGB37Y 45486011 Ki = 967 nM T60693 C1TJC6 45486012 Ki = 4568 nM T60693 CHQI57 45486013 Ki = 4595 nM T60693 C0KXD9 45486018 Ki = 2043 nM T60693 CF46MY 45486027 Ki = 98 nM T60693 C9DVC1 45486028 Ki = 726 nM T60693 C3EV6H 45486032 Ki = 508 nM T60693 CV1N7L 45486033 Ki = 1451 nM T60693 C9F4WP 45486035 Ki = 1358 nM T60693 CC6DZ4 45486042 Ki = 121 nM T60693 CE1MR2 45486046 Ki = 495 nM T60693 CW7I8C 45486055 Ki = 744 nM T60693 C5JE6L 45486062 Ki = 2191 nM T60693 CL2QF9 45486070 Ki = 263 nM T60693 CM39DL 45486096 Ki = 453 nM T60693 C60VCS 45486101 Ki = 726 nM T60693 CGY05X 45486102 Ki = 1189 nM T60693 C6YS7G 45486258 Ki = 26 nM T60693 C8CKM0 45487174 Ki = 15 nM T60693 CSC23N 45487200 Ki = 41 nM T60693 CFC45O 45487206 Ki = 1140 nM T60693 C3QU2C 45487384 IC50 > 5000 nM T60693 CO7VJ6 46190938 Ki = 45 nM T60693 CO0Z6H 46190939 Ki > 890 nM T60693 CV89LB 46226159 Ki > 890 nM T60693 COZ08F 46226176 Ki = 79 nM T60693 CL10HJ 46226250 Ki = 41 nM T60693 C7RL2Y 46227748 Ki = 10000 nM T60693 CT9AF7 46227758 Ki > 5000 nM T60693 CUK71N 46227759 Ki > 5000 nM T60693 C7JYA3 46227761 Ki > 10000 nM T60693 CKO64X 46227768 Ki = 22 nM T60693 CE4K7J 46227769 Ki = 674 nM T60693 C3YHF0 46227961 Ki = 0.015 nM T60693 C7LW1S 46227963 Ki = 0.34 nM T60693 C9L6WI 46227966 Ki = 0.37 nM T60693 C6RK5N 46230439 Ki = 2880 nM T60693 CSD7C9 46230440 Ki > 10000 nM T60693 CK4TO1 46230441 Ki = 2220 nM T60693 C7L1QA 46230532 Ki = 720 nM T60693 C5UZ4O 46230533 Ki = 10000 nM T60693 C2QE0Y 46230534 Ki = 3380 nM T60693 CDF6P8 46230535 Ki = 935 nM T60693 CC85FR 46237455 Ki > 1000 nM T60693 CMJ0K7 46237580 Ki = 920 nM T60693 C3R4KL 46237583 Ki > 1000 nM T60693 CC0K6V 46237584 Ki > 1000 nM T60693 CSH53K 46237585 Ki > 1000 nM T60693 CQ6K9E 46237703 Ki > 1000 nM T60693 C0G6MX 46237708 Ki = 70 nM T60693 CNC81F 46237832 Ki = 1510 nM T60693 C97MLP 46237834 Ki = 6 nM T60693 C45EPA 46237835 Ki = 850 nM T60693 CAY07H 46237836 Ki = 120 nM T60693 CCP98G 46237837 Ki > 1000 nM T60693 CIFP51 46245518 EC50 = 31 nM T60693 C30XLJ 46831301 Ki = 4.4 nM T60693 CK28BZ 46832153 Ki = 63 nM T60693 C8OK1P 46867404 EC50 = 6 nM T60693 C0J5XV 46867466 Ki = 0.617 nM T60693 C03LTM 46869265 Ki = 820000 nM T60693 CO5NQ3 46877612 Ki = 20.1 nM T60693 CF9G0A 46877633 Ki = 11 nM T60693 C5A7HD 46877642 Ki = 4.11 nM T60693 CVU37F 46877653 Ki = 0.7 nM T60693 CG19YU 46877660 Ki = 11.9 nM T60693 CJXS34 46877820 Ki = 61.4 nM T60693 C4R3BH 46877822 Ki = 1.4 nM T60693 CD16LI 46877823 Ki = 0.49 nM T60693 CFT4H0 46877824 Ki = 0.11 nM T60693 C57PVS 46877825 Ki = 0.37 nM T60693 CM89BU 46877826 Ki = 0.08 nM T60693 C6T7DS 46877827 Ki = 0.6 nM T60693 CK7CY0 46878243 Ki = 1.5 nM T60693 CUMN01 46878245 Ki = 5.5 nM T60693 CJR0C1 46878247 Ki = 0.57 nM T60693 C7HT9Q 46880391 Ki = 6.2 nM T60693 CARP46 46880392 Ki = 0.99 nM T60693 C12DCB 46880393 Ki = 0.17 nM T60693 C65ALC 46880394 Ki = 12 nM T60693 CKQ94Y 46880395 Ki = 9.8 nM T60693 C5HDU1 46880396 Ki = 3.3 nM T60693 C82AOZ 46880397 Ki = 3.9 nM T60693 CW3F8K 46880398 Ki = 1.4 nM T60693 CKJD61 46880399 Ki = 0.34 nM T60693 C1RZ7T 46880400 Ki = 36 nM T60693 CV7K6J 46880401 Ki = 8.3 nM T60693 C49NWA 46880452 Ki = 0.2 nM T60693 C7JK5C 46880453 Ki = 52 nM T60693 CE6Y5T 46880454 Ki = 22 nM T60693 CK8A1O 46880462 Ki > 10000 nM T60693 C9KDP4 46880463 Ki > 10000 nM T60693 CODR73 46880498 Ki > 10000 nM T60693 CHJ5Y6 46880566 Ki > 10000 nM T60693 CE9PG2 46880567 Ki > 10000 nM T60693 C01PGO 46880568 Ki > 10000 nM T60693 CS7L4X 46880569 Ki > 10000 nM T60693 C0PXY7 46880628 Ki > 10000 nM T60693 CD37LU 46880629 Ki > 10000 nM T60693 CUY89F 46880630 Ki > 10000 nM T60693 C4P6XS 46880631 Ki > 10000 nM T60693 CJ53KF 46880672 Ki > 10000 nM T60693 CYJC08 46880673 Ki > 10000 nM T60693 C1RI9O 46880674 Ki > 10000 nM T60693 COP1Z5 46906945 Ki = 15 nM T60693 CGM92J 46907011 Ki = 0.279 nM T60693 CQ5S8B 46907012 Ki = 0.135 nM T60693 CA3HM0 46907038 Ki = 39 nM T60693 C5ZDY3 46915370 Ki = 1800 nM T60693 C0YJ1U 46928474 Ki = 13 nM T60693 CQ86RS 46928475 Ki = 0.151 nM T60693 C0HQ9F 46928476 Ki = 13 nM T60693 CI86QW 46928478 Ki = 0.066 nM T60693 CR3O7S 46928581 Ki = 6.9 nM T60693 CV93BN 46945445 Ki > 10000 nM T60693 C0H1AC 46945446 Ki > 10000 nM T60693 CTKZ20 46994934 Ki = 3000 nM T60693 CV16YQ 47023707 Ki > 100000 nM T60693 CO1Q4L 47038967 Ki = 2290.87 nM T60693 CABL63 49765080 IC50 = 204 nM T60693 C2LZJ0 49783209 Ki > 10000 nM T60693 C57SMG 49783415 Ki > 10000 nM T60693 C0TG6I 49783419 Ki > 10000 nM T60693 CYP36E 49799951 Ki > 1000 nM T60693 CTR1Y2 49799964 EC50 = 13.9 nM T60693 CDS18H 49799966 Ki = 43.3 nM T60693 C4FA1V 49799967 Ki = 3.9 nM T60693 CEG52T 49799968 EC50 = 559 nM T60693 C2H8LY 49799969 EC50 = 2 nM T60693 C3T6NH 49843555 Ki > 577 nM T60693 CXW97O 49865703 IC50 = 1301 nM T60693 CRG60N 49865732 IC50 = 172 nM T60693 CZY2T3 49865733 Ki = 40 nM T60693 CI2W0D 49865783 IC50 = 596 nM T60693 CUK35O 49865784 IC50 = 338 nM T60693 CLD4P0 49865785 IC50 = 8242 nM T60693 CL0DR3 49865859 IC50 = 1489 nM T60693 CE15WQ 49865860 IC50 = 8624 nM T60693 C4EM1X 49865861 IC50 = 14161 nM T60693 CEF3O1 49865862 IC50 = 17802 nM T60693 C5YP2L 49865863 IC50 > 30000 nM T60693 CNGL32 49865918 IC50 > 30000 nM T60693 C9HEP1 49865919 IC50 = 222 nM T60693 CL6ZG8 49865920 IC50 = 1733 nM T60693 CC6VB8 49865921 IC50 = 3500 nM T60693 CHYN61 49865922 IC50 = 4176 nM T60693 C5NJ6K 49865969 IC50 > 30000 nM T60693 C3CJ4R 49865970 IC50 = 10729 nM T60693 CP8VQ6 49865971 IC50 = 462 nM T60693 CAI09G 49865972 IC50 = 2698 nM T60693 C5TMG9 49865973 IC50 = 19287 nM T60693 C87OZE 49866022 IC50 > 30000 nM T60693 CN7X5V 49866023 IC50 > 30000 nM T60693 C3L4OQ 49866024 IC50 > 30000 nM T60693 CFT26X 49866025 IC50 = 347 nM T60693 C2RY0J 50878551 Ki = 1122.02 nM T60693 C1W6TV 50898777 Ki > 10000 nM T60693 CXMZ73 50898778 Ki > 10000 nM T60693 CG4SX0 50942591 Ki = 42 nM T60693 C9Y5CM 50964436 Ki > 100000 nM T60693 CU63SQ 50994498 Ki = 372 nM T60693 C5D0NY 51002736 Ki = 225 nM T60693 C3OQP7 51002739 Ki = 367 nM T60693 CBPQ82 51002822 Ki = 210 nM T60693 CCTI18 51002823 Ki = 72 nM T60693 CFGZ31 51002824 Ki = 322 nM T60693 CSW52C 51002825 Ki = 475 nM T60693 C8OFC7 51002870 Ki = 125 nM T60693 CG7US6 51002874 Ki = 123 nM T60693 C0B8ZH 51002978 Ki = 323 nM T60693 C7FI2R 51002981 Ki = 390 nM T60693 C7QA4S 51003039 Ki = 174 nM T60693 CGU3H2 51003042 Ki = 153 nM T60693 C08HUZ 51003216 EC50 = 11 nM T60693 CXW86B 51003218 EC50 = 1.28 nM T60693 CW5Q7V 51003448 Ki = 316.23 nM T60693 CGR98N 51003449 Ki = 19.95 nM T60693 C9WEO3 51003467 Ki = 0.23 nM T60693 CNV2Q4 51004758 IC50 = 3410 nM T60693 C1SK7C 51009928 IC50 > 10000 nM T60693 CM2K7S 51042171 Ki > 10000 nM T60693 CE4KP1 51050257 Ki > 10000 nM T60693 C32GVN 51051674 Ki = 2600 nM T60693 C17BSI 51051707 Ki = 229.09 nM T60693 CQ6SR3 51353734 Ki = 3.7 nM T60693 CDQ3I6 51353736 Ki = 0.71 nM T60693 C4GH6F 51353738 Ki = 5.8 nM T60693 CZ1CL5 51353740 Ki = 11 nM T60693 C3W7AJ 51353742 Ki = 1.2 nM T60693 CK07VQ 51353744 Ki = 0.94 nM T60693 C9JAE4 51356293 Ki = 0.3 nM T60693 C7MNL4 51356294 Ki = 0.83 nM T60693 C3S0LD 51356295 Ki = 0.84 nM T60693 C6OY1E 51356296 Ki = 4.8 nM T60693 C54EPI 51356297 Ki = 2.1 nM T60693 CAU84H 51356590 Ki = 3.5 nM T60693 CZ1GB9 51356591 Ki = 18 nM T60693 CE16YQ 51356593 Ki = 21 nM T60693 CGF0L6 51356594 Ki = 95 nM T60693 CY5A7R 51357141 Ki = 2.4 nM T60693 CQ5Y6C 51357143 Ki = 1.6 nM T60693 CYB1A0 51357420 Ki = 0.45 nM T60693 C38DJS 52210045 Ki = 2930 nM T60693 C0TCI3 52915030 IC50 = 1269 nM T60693 CK6GN5 52915031 IC50 = 1049 nM T60693 CXF14W 52915032 IC50 = 900 nM T60693 C27KOF 52915269 IC50 = 3079 nM T60693 CQ71YX 52915270 IC50 = 5924 nM T60693 CH56XF 52915389 IC50 = 3669 nM T60693 C02UBO 52915390 IC50 = 1157 nM T60693 CP2M6E 52915391 IC50 = 1850 nM T60693 CPA43I 52915392 IC50 = 4955 nM T60693 C5OA9H 52915393 IC50 = 2565 nM T60693 CA3P2C 52915514 IC50 = 4348 nM T60693 CK39TQ 52915515 IC50 = 1649 nM T60693 C98UZW 52915516 IC50 = 4257 nM T60693 CLAS61 52915517 IC50 = 2155 nM T60693 C7FDE9 52915518 IC50 = 1222 nM T60693 C9YOD2 52915634 IC50 = 998 nM T60693 C1ZHF3 52915635 IC50 = 872 nM T60693 CZB67C 52915636 IC50 = 6177 nM T60693 CE3IS2 52915637 IC50 = 9103 nM T60693 CYB6J8 52916598 IC50 = 5475 nM T60693 CG1F9W 52916599 IC50 = 1091 nM T60693 C7NO2D 52916712 IC50 = 1496 nM T60693 CZ3K9S 52916713 IC50 = 1347 nM T60693 CI32WO 52916714 IC50 = 1023 nM T60693 C09MKV 52940733 Ki > 1000 nM T60693 C1M3SD 52941462 IC50 = 754 nM T60693 C58ART 52941549 IC50 = 1126 nM T60693 C7Z4OK 52942515 Ki > 1000 nM T60693 CYLC29 52942529 IC50 = 46 nM T60693 CPOQ82 52942580 IC50 = 3159 nM T60693 C3YF5D 52942581 IC50 = 6691 nM T60693 CX5F9O 52942614 Ki = 24.3 nM T60693 CKN2U6 52942810 IC50 = 1410 nM T60693 C5V4DW 52943162 IC50 = 49 nM T60693 C3QLR8 52943731 Ki = 197 nM T60693 CNK14O 52943803 IC50 = 11 nM T60693 CLU6S9 52943962 Ki = 146 nM T60693 CRH1Q5 52943993 IC50 = 24234 nM T60693 CBW0A9 52944041 IC50 = 20502 nM T60693 C89GIK 52944552 IC50 = 431 nM T60693 CP5A3T 52944907 IC50 = 683 nM T60693 C54ZBG 52944974 IC50 = 130 nM T60693 CV48KS 52945118 IC50 = 345 nM T60693 C1G0IP 52945138 IC50 = 1003 nM T60693 CSZ4R3 52945588 IC50 = 342 nM T60693 CBO48U 52945590 EC50 = 239 nM T60693 CNGU78 52945626 IC50 = 148 nM T60693 CG8CN4 52946340 IC50 = 3411 nM T60693 C1V8ET 52947396 Ki > 1000 nM T60693 CFD18K 52947437 IC50 = 12589 nM T60693 CFN7I8 52947509 IC50 = 90 nM T60693 CYIX94 52947511 Ki = 422 nM T60693 C41AYU 52947523 IC50 = 524 nM T60693 CY06OH 52947573 IC50 = 355 nM T60693 CY72CQ 52947593 IC50 = 846 nM T60693 CFI96N 52947735 IC50 = 620 nM T60693 CI63UL 52948240 IC50 = 241 nM T60693 CAID24 52948615 Ki = 0.5 nM T60693 C15KNW 52948655 IC50 = 307 nM T60693 C48RBH 52948719 IC50 = 215 nM T60693 CZX5B9 52948735 IC50 = 39 nM T60693 CE0R3S 52948850 IC50 = 13266 nM T60693 CPN4Z8 52948969 IC50 = 111 nM T60693 CZX6F9 52949241 Ki = 198 nM T60693 CVWY23 52949439 IC50 = 386 nM T60693 C9V6GB 52950007 IC50 = 2193 nM T60693 CPA2G4 52951481 Ki = 798 nM T60693 CYP0I3 52951482 Ki = 597 nM T60693 C01KMG 52952006 Ki = 120 nM T60693 CL1QG4 52952007 Ki = 60 nM T60693 CET8Q0 52952008 Ki = 790 nM T60693 C6X7WL 52952107 Ki > 13000 nM T60693 C4N9HF 52952108 Ki = 290 nM T60693 CWC1N8 52952109 Ki = 228 nM T60693 C7JB4Q 52952110 Ki = 286 nM T60693 C2GPE5 52952207 Ki > 8000 nM T60693 CTU43X 53316968 Ki = 387 nM T60693 CCOD69 53316969 EC50 = 194 nM T60693 CE3P7Y 53317205 Ki = 794.33 nM T60693 C0NKY7 53317262 Ki = 630.96 nM T60693 C7H8QK 53318490 Ki > 3981.07 nM T60693 C31ZOA 53318757 Ki = 630.96 nM T60693 CI6CQ0 53319615 Ki > 570 nM T60693 C6SY4G 53319616 Ki > 570 nM T60693 CB10OV 53319822 Ki = 25.12 nM T60693 CT8R3I 53319870 Ki = 630.96 nM T60693 C4XD5Q 53319871 Ki = 199.53 nM T60693 CY5MG9 53321111 Ki = 1258.93 nM T60693 CD14AE 53321176 Ki > 3981.07 nM T60693 C6X9OT 53321653 Ki > 3981.07 nM T60693 C2EV1S 53322245 Ki = 275 nM T60693 C1L8IV 53322246 Ki > 570 nM T60693 CRN26Z 53322438 Ki = 316.23 nM T60693 CZY2G3 53322439 Ki = 630.96 nM T60693 CMOL62 53322496 Ki = 199.53 nM T60693 CLDI90 53323074 Ki = 12 nM T60693 C30TBO 53323800 Ki = 1000 nM T60693 CS9I6Z 53323801 Ki = 630.96 nM T60693 CGI94L 53323802 Ki = 125.89 nM T60693 C5I4KQ 53323803 Ki = 251.19 nM T60693 C0ZJ1T 53323804 Ki = 158.49 nM T60693 CV5EC1 53323805 Ki = 199.53 nM T60693 C7Z4KR 53323841 Ki > 3981.07 nM T60693 C32YWL 53324045 Ki = 1328 nM T60693 CJ59GU 53325079 Ki = 63.1 nM T60693 CH37ZT 53325227 Ki = 3784 nM T60693 CRQF15 53325242 Ki = 2669 nM T60693 C5E7LW 53325608 EC50 = 18 nM T60693 CL5WG8 53325725 Ki = 1.4 nM T60693 CRZ76L 53326167 Ki = 39 nM T60693 CLP1Q0 53326367 Ki = 501.19 nM T60693 C7ETI8 53326368 Ki = 1258.93 nM T60693 CI3K7N 53326835 Ki = 251.19 nM T60693 CA3KL4 53388149 EC50 = 26.4 nM T60693 C0TIQ5 53388316 EC50 = 25 nM T60693 CKIU81 53388785 IC50 = 32400 nM T60693 CFE6S4 53465409 Ki = 10 nM T60693 CT62EG 53465411 Ki = 25 nM T60693 CU04GB 53465412 Ki = 75 nM T60693 C7V4ME 53465413 Ki = 33 nM T60693 C89NMJ 53465486 Ki = 14 nM T60693 CDV57J 53465487 Ki = 2.2 nM T60693 CN2P0M 53465488 Ki = 5.8 nM T60693 C03LXZ 53465489 Ki = 13 nM T60693 C7JV2P 53465490 Ki = 1.8 nM T60693 C0NW4J 53465491 Ki = 3.7 nM T60693 C6C1FN 53465556 Ki = 1.1 nM T60693 CQ5F0H 53465557 Ki = 54 nM T60693 CW8XR1 53465558 Ki = 72 nM T60693 CL27OF 53465559 Ki = 8.8 nM T60693 CB7F1V 53465560 Ki = 157 nM T60693 CF87WN 53465561 Ki = 84 nM T60693 CJX6G9 53465633 Ki = 66 nM T60693 C5W8PL 53465634 Ki = 26 nM T60693 CR8FE6 53465635 Ki = 584 nM T60693 CBFI98 53465636 Ki = 75 nM T60693 C6MS1K 53465637 Ki > 222 nM T60693 CUR52F 53465638 Ki = 54 nM T60693 CI18GY 53465639 Ki = 53 nM T60693 C8D7CS 53465710 Ki = 8.4 nM T60693 CR1VM6 53466534 Ki = 62 nM T60693 CMOZ61 53475319 Ki > 10000 nM T60693 CO8ZP9 53498895 Ki = 11100 nM T60693 CFU5Q7 53619719 Ki = 676.08 nM T60693 C70BZV 54580938 Ki = 0.073 nM T60693 CYEC84 54581367 Ki = 110 nM T60693 C3I0HF 54582933 Ki = 0.28 nM T60693 C9G8RT 54582934 Ki = 0.37 nM T60693 CX0O1G 54583374 Ki = 6.4 nM T60693 CHA7T8 54584041 Ki = 0.23 nM T60693 C96ISF 54584882 Ki = 0.2 nM T60693 CKUH91 54585844 Ki = 0.14 nM T60693 C6MHV9 54585845 Ki = 0.27 nM T60693 CV86NQ 54586810 Ki = 0.37 nM T60693 CQ83TL 54596311 Ki = 5430 nM T60693 C3EP9X 54669894 Ki > 1000000 nM T60693 CXF1G9 54751920 Ki > 100000 nM T60693 CNT03F 54754507 Ki > 100000 nM T60693 CROS84 54756989 Ki = 1.59 nM T60693 C2ISE6 54756990 EC50 = 0.88 nM T60693 C7F6EC 54757387 Ki > 1000000 nM T60693 CQU87I 56589659 EC50 = 39.8 nM T60693 CHZ1D7 56589680 EC50 = 307 nM T60693 CP5R4Y 56595310 Ki > 10000 nM T60693 C28AED 56655502 Ki = 0.565 nM T60693 CP5E2J 56657871 Ki = 55 nM T60693 CCN2E8 56658044 EC50 = 5.33 nM T60693 CJW5C1 56658452 Ki = 19.9 nM T60693 CP37LM 56659141 Ki = 4.7 nM T60693 C69VIF 56661555 Ki = 45.6 nM T60693 CJ2MA7 56663008 Ki = 0.08 nM T60693 CDKP63 56664973 Ki = 5.63 nM T60693 C2KG9D 56665110 Ki = 662.4 nM T60693 CEW3K4 56665405 Ki = 1.65 nM T60693 CR64WX 56665407 Ki = 9.01 nM T60693 C3QLV1 56666529 Ki = 367 nM T60693 C4QM3N 56668405 Ki = 9.93 nM T60693 C8O7MT 56668839 Ki = 0.15 nM T60693 CL21RS 56669900 Ki = 9 nM T60693 CO18SG 56669938 Ki > 8600 nM T60693 C9SY1A 56672310 Ki = 0.58 nM T60693 C2NQJ4 56673010 Ki = 2.49 nM T60693 CD9JK4 56675713 Ki = 2.83 nM T60693 CG1XO8 56676328 Ki = 9 nM T60693 C45KMW 56676759 Ki = 7500 nM T60693 C0WVZ6 56676760 Ki = 171 nM T60693 CVXJ29 56676761 Ki = 98 nM T60693 CQZ75Y 56678873 Ki = 1230 nM T60693 CZ6B0O 56678874 Ki = 51 nM T60693 C15FOK 56679008 Ki = 0.18 nM T60693 CDG30L 56680069 Ki = 199 nM T60693 CX8F2N 56681954 Ki = 8.92 nM T60693 C2A4MQ 56681955 Ki = 35.5 nM T60693 CP3L7E 56682094 Ki = 1203 nM T60693 CK52GV 56682330 Ki = 6.49 nM T60693 CJ19ZL 56787422 Ki = 151.36 nM T60693 CHON57 56807426 Ki = 2570.4 nM T60693 C95LAM 56834761 Ki > 1000000 nM T60693 CRX31L 56840667 Ki = 918 nM T60693 CQ2O4U 56849549 Ki = 1.41 nM T60693 CCMS01 56849550 Ki = 1.05 nM T60693 C7VT5K 56849551 Ki = 26.7 nM T60693 C2Y9CE 56851423 Ki = 9.21 nM T60693 C34PMD 56851424 Ki = 1.49 nM T60693 CN32ZB 56851582 Ki = 0.622 nM T60693 CY9DH2 56851583 Ki = 0.722 nM T60693 CC3JS8 56851584 Ki = 44.9 nM T60693 C9E6CU 56851585 Ki = 53.7 nM T60693 C1ZOM5 56851586 Ki = 14 nM T60693 C1RDE6 56892310 Ki = 346.74 nM T60693 CK3WH4 56951181 Ki = 2.5 nM T60693 CS1K0A 57391716 Ki = 604 nM T60693 CJ38ZY 57393448 Ki = 483 nM T60693 CS02AB 57395174 Ki = 3800 nM T60693 C3BR0J 57396943 Ki = 8300 nM T60693 C12ASH 57396944 Ki = 140 nM T60693 C3QF9I 57401062 Ki = 2.36 nM T60693 CDZ04Q 57401743 Ki = 40 nM T60693 C8RX7I 57402172 Ki = 751 nM T60693 CUL3W2 57402462 Ki = 419 nM T60693 CE46KV 57403475 Ki = 18 nM T60693 CT1IN3 57412337 Ki = 8.5 nM T60693 C7F4PN 57412339 Ki = 27 nM T60693 CTO37U 57412341 Ki = 23 nM T60693 C0UZ3G 57412343 Ki = 4.1 nM T60693 C3JL0D 57412421 Ki = 500 nM T60693 C10ZIE 57412591 Ki = 370 nM T60693 C8A1JR 57412593 Ki = 220 nM T60693 C5Q7KD 57412595 Ki = 910 nM T60693 C2WG9D 57412599 Ki = 560 nM T60693 C5D6QU 57412771 Ki = 0.99 nM T60693 CNI7Y9 57412772 Ki = 2.2 nM T60693 C21LRT 57412773 Ki = 3.5 nM T60693 CFB58K 57412848 Ki = 4.5 nM T60693 CTV4X5 57412849 Ki = 4.5 nM T60693 CSYI37 57412850 Ki = 1.1 nM T60693 CJI87G 57412851 Ki = 1.3 nM T60693 CCB0G9 57412852 EC50 = 0.43 nM T60693 CDV4H9 57412853 EC50 = 0.077 nM T60693 CAO20P 57412942 EC50 = 0.79 nM T60693 CF1LC3 57412943 Ki = 1.7 nM T60693 CYN92K 57412944 Ki = 1.9 nM T60693 C54XQG 57412945 Ki = 2.3 nM T60693 C0GL5A 57412946 Ki = 0.26 nM T60693 CGN29J 57413036 Ki = 0.36 nM T60693 C5ZHT6 57413037 Ki = 0.27 nM T60693 CP9L1N 57413038 Ki = 10 nM T60693 CP6G5F 57413039 Ki = 19 nM T60693 CH0B1F 57413040 Ki = 25 nM T60693 C0J3LY 57900041 Ki = 2.2 nM T60693 C6AWU4 57900045 Ki = 1.4 nM T60693 CY1TN7 57978734 Ki > 1000 nM T60693 C7MI3X 58046500 Ki = 80 nM T60693 CFXC84 58046524 Ki = 70 nM T60693 CI5H3N 58268566 Ki > 375 nM T60693 C6Z9JF 58268629 Ki > 400 nM T60693 C7EFU5 58443192 Ki = 1.6 nM T60693 C73BYR 58443217 EC50 = 0.62 nM T60693 C5V8NC 58443218 Ki = 1.3 nM T60693 C7Z8SF 58443225 Ki = 0.49 nM T60693 CS70GT 58443229 Ki = 3.3 nM T60693 CFXB82 58443230 Ki = 2.4 nM T60693 C4FKN0 58443234 EC50 = 0.34 nM T60693 CW81HV 58443235 Ki = 1.8 nM T60693 C6GA5O 60150457 Ki = 40 nM T60693 C7N0KO 60150458 EC50 = 12.2 nM T60693 C6G5TY 60154189 Ki > 400 nM T60693 C8MS6N 60154191 Ki > 400 nM T60693 CW63KM 60154192 Ki > 400 nM T60693 C2QX6R 60154193 Ki > 400 nM T60693 CD46EJ 60154264 Ki > 400 nM T60693 CEB0P5 60166738 Ki = 1566 nM T60693 C95OTB 62350121 Ki = 154.88 nM T60693 C7KLB6 68196155 EC50 = 1 nM T60693 CN1YW0 68642339 IC50 = 1200 nM T60693 CYBC09 68775633 Ki = 22 nM T60693 CCK5Z9 68776073 EC50 = 33 nM T60693 CHF83Z 68776748 EC50 = 330 nM T60693 CJAH92 68777672 EC50 = 20 nM T60693 CA56LT 68777734 EC50 = 600 nM T60693 CKX63G 68777945 EC50 = 220 nM T60693 CVF8G6 68778394 EC50 = 56 nM T60693 C1I8MB 68778890 EC50 = 26 nM T60693 C27KQI 68779363 EC50 = 41 nM T60693 C83YWM 68779815 EC50 = 12 nM T60693 CK4MH1 68782313 EC50 = 260 nM T60693 C89TSB 68867300 Ki = 0.12 nM T60693 C4DO7H 70158365 Ki > 890 nM T60693 C30HMT 70681352 Ki = 8470 nM T60693 CS1E7F 70681353 Ki = 2260 nM T60693 C9AW5C 70682920 Ki > 1000 nM T60693 C5JLS9 70683421 Ki = 30 nM T60693 CJ79UV 70683422 Ki > 10000 nM T60693 CH64DO 70683436 Ki = 110 nM T60693 CZW6K5 70683437 Ki = 9210 nM T60693 CX3M0F 70683438 Ki = 320 nM T60693 CXY52W 70685543 Ki = 220 nM T60693 C60FVD 70685544 Ki = 31 nM T60693 CU7V8F 70685545 Ki > 10000 nM T60693 CRKY09 70685720 IC50 = 3.07 nM T60693 CQL0S6 70687673 Ki = 1120 nM T60693 CY8DQ1 70687674 Ki = 1070 nM T60693 CE6K8V 70687698 Ki = 500 nM T60693 C3J5XF 70688073 EC50 = 1480 nM T60693 C1SH5O 70688074 EC50 = 176 nM T60693 CS86LY 70689742 Ki > 10000 nM T60693 C8B7ES 70691647 Ki = 0.11 nM T60693 CCQ5Z6 70691889 Ki > 10000 nM T60693 CR0G1C 70692260 EC50 = 3 nM T60693 C1A7LO 70693567 EC50 = 20.9 nM T60693 C9PQ4F 70693930 Ki = 150 nM T60693 CWO5F0 70695375 Ki > 400 nM T60693 CRG52J 70695535 Ki > 10000 nM T60693 C2V8UI 70696034 Ki = 290 nM T60693 CG3U7F 70697391 Ki > 400 nM T60693 CKD60A 70789640 Ki = 1208 nM T60693 CJ5DI4 70822235 Ki = 4.33 nM T60693 CI8M5U 70834572 Ki = 4070 nM T60693 CLQ46F 71155070 Ki = 776 nM T60693 C3XUP4 71155072 Ki = 7100 nM T60693 CXM90F 71155076 Ki = 93.4 nM T60693 CEOQ43 71229805 Ki = 0.044 nM T60693 CIK86Q 71230334 EC50 = 1.09 nM T60693 CLA6O8 71449105 IC50 = 2970 nM T60693 C2TY6U 71449133 Ki = 1.82 nM T60693 CEB0P4 71449173 IC50 = 5740 nM T60693 C8HV9A 71449570 Ki > 5000 nM T60693 CYG07C 71449995 Ki = 0.13 nM T60693 CK69PO 71450043 Ki = 1.21 nM T60693 C4TVF1 71450063 Ki > 100000 nM T60693 CHQZ46 71450134 Ki = 5.97 nM T60693 CSC3R7 71450213 Ki = 10.9 nM T60693 C9VZ8J 71450550 Ki = 1107 nM T60693 CJL59V 71450766 Ki = 0.45 nM T60693 C4BP5T 71450767 Ki = 0.2 nM T60693 CQ6M2A 71450900 IC50 = 1710 nM T60693 C6ZX3S 71450925 Ki = 23.7 nM T60693 C5YIC1 71450926 Ki = 29.8 nM T60693 C2R7GS 71450927 Ki = 9.95 nM T60693 CMB7X9 71450932 Ki = 36.1 nM T60693 CNP02X 71450939 EC50 = 0.8 nM T60693 C08KHB 71452040 Ki = 5.9 nM T60693 C0XW8E 71452041 Ki = 0.49 nM T60693 C20RPJ 71452224 EC50 = 25 nM T60693 C4NDR3 71452382 Ki = 1575 nM T60693 CDTW09 71452387 Ki = 1426 nM T60693 CYU3K7 71452742 Ki = 0.13 nM T60693 C4B6HU 71452746 Ki = 63.8 nM T60693 CYFH30 71452786 IC50 = 7560 nM T60693 CQY10P 71453677 Ki = 4.28 nM T60693 CRY4A1 71453704 Ki > 100000 nM T60693 CYOS40 71453706 Ki > 100000 nM T60693 CW0H5Q 71453774 Ki = 112 nM T60693 CZ08WY 71454361 EC50 = 0.26 nM T60693 CG82PA 71454362 Ki = 1.3 nM T60693 CM0H5E 71454460 Ki = 372 nM T60693 CXQ1G0 71454513 Ki = 21 nM T60693 CGM86O 71454514 Ki = 1.72 nM T60693 CQ5JE8 71454515 Ki = 26.4 nM T60693 CI16ON 71454516 Ki = 67.9 nM T60693 CO01LV 71454517 Ki = 0.52 nM T60693 C09IMN 71454521 Ki > 1900 nM T60693 CCKA54 71454553 IC50 > 10000 nM T60693 CYJ9X8 71454554 IC50 > 10000 nM T60693 CN3EX8 71455429 Ki > 100000 nM T60693 CW63BC 71455505 Ki = 3.31 nM T60693 C89UMR 71455506 Ki = 1.55 nM T60693 C6G2HC 71455894 Ki = 1147 nM T60693 CFBC49 71455896 Ki = 2688 nM T60693 C83WJY 71456105 Ki = 5.2 nM T60693 CQ0UG3 71456106 EC50 = 0.086 nM T60693 CF9HA1 71456174 Ki = 0.1698 nM T60693 C8FXZ5 71456257 Ki = 7.79 nM T60693 CDQM86 71456258 EC50 = 56.9 nM T60693 CXZ2V8 71456262 EC50 = 0.1 nM T60693 C42MER 71457207 Ki = 33000 nM T60693 C3XIP8 71457209 Ki > 100000 nM T60693 C9UVJ1 71457210 Ki > 100000 nM T60693 CLN75C 71457288 Ki = 5.37 nM T60693 CH4Y5I 71457289 Ki = 27.99 nM T60693 CPUO14 71457290 Ki = 3.1 nM T60693 C4KD6E 71457291 Ki = 12 nM T60693 C0R8UO 71457292 Ki = 4.41 nM T60693 CDSX56 71457372 Ki = 141 nM T60693 CP7JI0 71457691 Ki = 1094 nM T60693 C9GQO5 71458037 IC50 > 10000 nM T60693 CSJ4A1 71458063 Ki = 3.11 nM T60693 CG98LJ 71458064 Ki = 1.41 nM T60693 CP6DQ7 71458116 IC50 = 9440 nM T60693 C92YCB 71458142 IC50 > 10000 nM T60693 C8LNZ6 71459067 Ki > 100000 nM T60693 CK5T4P 71459604 Ki = 1420 nM T60693 C7X9YH 71459820 Ki = 2.7 nM T60693 CA1N5D 71459821 Ki = 1.3 nM T60693 CTWI83 71459939 Ki = 24.9 nM T60693 CQ52LR 71459947 Ki = 22.2 nM T60693 CFR1T9 71459948 Ki = 155 nM T60693 CUID52 71459949 Ki = 44.7 nM T60693 C0TP7N 71459950 Ki = 109 nM T60693 CHS4D2 71459951 Ki = 1.85 nM T60693 CE2VA0 71459952 EC50 = 1.78 nM T60693 CBHT09 71459962 EC50 = 0.1 nM T60693 C6NOP7 71459993 IC50 > 10000 nM T60693 C6IG5K 71460019 IC50 > 10000 nM T60693 C12KHQ 71460850 Ki = 1.57 nM T60693 CJ65RV 71460942 Ki = 1.82 nM T60693 CC25XY 71460943 Ki = 49 nM T60693 CT52OM 71460944 Ki = 1.53 nM T60693 C6NLR9 71460945 Ki = 17 nM T60693 CBEV63 71461579 Ki = 318 nM T60693 CV60JN 71461663 Ki = 159 nM T60693 CFHE81 71461664 Ki = 58 nM T60693 CXT37B 71461665 Ki = 5.3 nM T60693 CY28RA 71461666 Ki = 1.64 nM T60693 C9Q6GY 71461668 Ki = 63.3 nM T60693 CD4Q0A 71461673 EC50 = 0.61 nM T60693 C6N1FP 71462554 Ki = 0.46 nM T60693 C4ZD8G 71462655 Ki = 5.33 nM T60693 CB3L8W 71462656 Ki = 117 nM T60693 CKX5O8 71463061 Ki = 2080 nM T60693 C1Y9IC 71463063 Ki = 617 nM T60693 C2I5MZ 71463280 Ki = 0.38 nM T60693 C79HRU 71473391 EC50 > 50000 nM T60693 C1C7OB 71499035 Ki = 420 nM T60693 CW8ZV5 71509717 EC50 = 50 nM T60693 C5OMH4 71516215 EC50 = 76 nM T60693 C7A1GD 71583623 Ki = 25 nM T60693 C0SL2D 71583625 Ki = 54 nM T60693 C8GVL2 71583725 Ki = 1.2 nM T60693 CAI8C4 71583726 Ki = 1200 nM T60693 CZ16QP 71583727 Ki = 130 nM T60693 CZF0O5 71583728 Ki = 110 nM T60693 C9Z7AT 71605588 Ki = 174 nM T60693 CG8ZD6 71605589 Ki = 205 nM T60693 CU53FL 71605755 Ki = 240 nM T60693 CMZ8F3 71605756 Ki = 180 nM T60693 CIW95L 71613507 Ki = 2 nM T60693 C26ORE 71613508 Ki = 21 nM T60693 CHI7D3 71613509 Ki = 148 nM T60693 CEO5Z2 71613709 Ki = 36 nM T60693 C8X6TP 71613710 Ki = 437 nM T60693 C82MIG 71613711 Ki = 302 nM T60693 C0MC1V 71613712 Ki = 575 nM T60693 CVC5H1 71613903 Ki = 263 nM T60693 CX9PM4 71613904 Ki > 10000 nM T60693 C2BOG7 71613905 Ki = 39 nM T60693 CAJ61F 71613906 Ki = 427 nM T60693 CS3CN1 71613907 Ki = 2291 nM T60693 C0B7LC 71624265 Ki = 190.2 nM T60693 C7Q9VU 71624266 Ki = 159.7 nM T60693 CXZ6E1 71624268 Ki = 43.9 nM T60693 C0O6IR 71624269 Ki = 29.2 nM T60693 CW2G0T 71624270 Ki = 41.77 nM T60693 CBM1C8 71624387 Ki = 39.2 nM T60693 CML7K2 71624388 Ki = 43.4 nM T60693 C1B9VM 71624389 Ki = 27.69 nM T60693 CA70EB 71624445 Ki = 0.051 nM T60693 CH3M7S 71624446 EC50 = 0.057 nM T60693 CJ2Z3X 71624447 Ki = 0.06 nM T60693 C5N9VQ 71624552 EC50 = 0.011 nM T60693 C86LGF 71624553 EC50 = 0.027 nM T60693 CC2O6N 71624554 EC50 = 0.031 nM T60693 CHUK68 71624555 EC50 = 0.017 nM T60693 CTBQ82 71624556 EC50 = 0.041 nM T60693 C5GY3N 71624661 EC50 = 0.068 nM T60693 CSRM32 71624662 EC50 = 0.071 nM T60693 C8PY7O 71624663 EC50 = 0.016 nM T60693 CO5FY6 71624665 Ki = 0.11 nM T60693 CG43FE 71624776 Ki = 0.15 nM T60693 CL1D9K 71624777 EC50 = 0.083 nM T60693 C1PCL3 71624778 Ki = 0.22 nM T60693 C5CYQ7 71624779 Ki = 0.16 nM T60693 CU3P1N 71624892 Ki = 0.11 nM T60693 CRAJ73 71624894 Ki = 0.067 nM T60693 C8D4NE 71624895 Ki = 0.059 nM T60693 CI86RQ 71625025 Ki = 0.078 nM T60693 C6DGY1 71625026 EC50 = 0.053 nM T60693 C6BHJ1 71625027 Ki = 0.015 nM T60693 CD28YT 71625028 Ki = 0.019 nM T60693 CMG6J7 71625029 Ki = 0.02 nM T60693 CFC4W3 71625148 Ki = 0.033 nM T60693 CDX2J0 71625149 Ki = 0.025 nM T60693 C4C2KN 71625150 EC50 = 0.035 nM T60693 C40NIQ 71625151 EC50 = 0.013 nM T60693 CN9OL5 71625152 EC50 = 0.0061 nM T60693 CTB9K7 71625277 EC50 = 0.007 nM T60693 CY8J0P 71625278 EC50 = 0.0077 nM T60693 CA4EU5 71625279 EC50 = 0.0098 nM T60693 C8KTI0 71625280 EC50 = 0.029 nM T60693 CA5W3M 71625281 EC50 = 0.047 nM T60693 C3ZX5Y 71625393 EC50 = 0.02 nM T60693 CC6J7G 71625394 Ki = 0.041 nM T60693 C4FO0S 71625395 Ki = 0.047 nM T60693 C1A9BS 71660039 Ki = 2882 nM T60693 CE0AX8 71660040 Ki = 238 nM T60693 CE5J8U 71660041 Ki = 163 nM T60693 CF4NS6 71660042 Ki = 71 nM T60693 CWBH85 71660081 Ki = 4182 nM T60693 CWKO96 71660082 Ki = 1651 nM T60693 CXZ1D7 71660083 Ki = 1913 nM T60693 CJK9R5 71660084 Ki = 971 nM T60693 C7R1TA 71660085 Ki = 2879 nM T60693 C4U5ZF 71660086 Ki = 2217 nM T60693 C64TPF 71660087 Ki = 730 nM T60693 CM6I2K 71660088 Ki = 670 nM T60693 CD9CN8 71660125 Ki = 721 nM T60693 CDS7T3 71660126 Ki = 826 nM T60693 C1AIY3 71660127 Ki = 2459 nM T60693 CJ43VK 71660128 Ki = 16 nM T60693 CF57LR 71660129 Ki = 80 nM T60693 C58SAC 71660130 Ki = 1922 nM T60693 CG7UJ9 71660163 Ki = 541 nM T60693 C5XM1H 71680922 Ki = 0.36 nM T60693 CUW3Z8 71680923 Ki = 0.16 nM T60693 CWSC46 71680924 Ki = 0.33 nM T60693 CP5FK9 71681076 Ki = 0.27 nM T60693 C4LV9A 71681077 Ki = 0.26 nM T60693 CE0YC8 71681078 Ki = 0.13 nM T60693 CU57ZQ 71681079 Ki = 0.33 nM T60693 CL6B7A 71716141 EC50 = 2.721 nM T60693 CVM39A 71716193 Ki = 0.5 nM T60693 C9F5QJ 71717732 EC50 = 0.051 nM T60693 CX9PV1 71717968 EC50 = 22.41 nM T60693 C7ZI9Q 71717970 EC50 = 3.787 nM T60693 CXE2V6 71718580 EC50 = 32.21 nM T60693 C4LI1B 71718582 EC50 = 11.26 nM T60693 C8QO1W 71719108 Ki = 948 nM T60693 CZ8CL2 71719454 Ki = 200 nM T60693 CPO6T5 71719795 EC50 = 8.071 nM T60693 C3LUG2 71720208 Ki = 8.33 nM T60693 CTU9Q8 71720326 IC50 = 7.7 nM T60693 C17DZG 71720406 EC50 = 2.231 nM T60693 CRO30V 71720457 Ki = 17 nM T60693 CY89EO 71720682 Ki = 192 nM T60693 CCB3X2 71726555 Ki = 14 nM T60693 C4G5IU 71726685 Ki = 3.5 nM T60693 CLBE62 71726686 Ki = 13 nM T60693 C0V9IX 71746034 Ki > 5000 nM T60693 CU47GC 71751564 Ki = 2 nM T60693 C0L7TE 71769137 Ki > 10000 nM T60693 CTX84S 71769138 Ki > 10000 nM T60693 C3YAR9 71769139 Ki > 10000 nM T60693 CWK9E7 71769267 Ki = 21000 nM T60693 C7G3EX 71769268 Ki > 10000 nM T60693 CEZW27 71769269 Ki = 2200 nM T60693 CW95UP 71819400 EC50 = 25000 nM T60693 C0EBP2 71819401 EC50 = 1600 nM T60693 C7SQL1 71819402 EC50 = 50000 nM T60693 C8HK9Y 71819403 EC50 = 126000 nM T60693 CW0YD6 71819525 EC50 = 32000 nM T60693 CILA50 71861855 Ki = 562.34 nM T60693 C0XHE7 72151344 Ki = 14400 nM T60693 C2QS5M 72153748 Ki = 5560 nM T60693 CQHB67 72202465 Ki = 3544 nM T60693 CZQ86Y 72374835 Ki = 1229 nM T60693 CAK42B 72374836 Ki = 135 nM T60693 CWH6T3 72548703 IC50 = 1.1 nM T60693 C7NB1W 72711408 Ki = 0.17 nM T60693 C89COK 72711409 Ki = 9 nM T60693 C7FI6P 72711410 Ki = 3.6 nM T60693 C29YGC 72712370 EC50 = 900 nM T60693 CYEJ30 72713098 Ki = 20.92 nM T60693 CJT7L9 72713099 Ki = 8.22 nM T60693 C4MWE1 72713100 Ki = 1.4 nM T60693 CPY8F1 72713101 Ki = 13.67 nM T60693 CBVG86 72713102 Ki = 9.9 nM T60693 CLRX12 72713104 Ki = 0.92 nM T60693 CC6Q5R 72771081 Ki < 100 nM T60693 C1UE4T 73212366 Ki = 310 nM T60693 C2A7EK 73212367 Ki = 140 nM T60693 C3J7AV 73212368 Ki = 110 nM T60693 CZU17T 73212369 Ki = 250 nM T60693 C4KF1I 73212370 Ki = 78 nM T60693 CIX34M 73212442 Ki = 330 nM T60693 C9EIS4 73212443 Ki = 150 nM T60693 C41NSY 73212444 Ki = 78 nM T60693 CGN9Q8 73212445 Ki = 89 nM T60693 COM5T7 73212446 Ki = 54 nM T60693 CB3M2F 73212447 Ki = 39 nM T60693 C0PTG7 73212818 EC50 = 1.3 nM T60693 CVC29M 73212819 EC50 = 16 nM T60693 CM8PD9 73212820 EC50 = 6.7 nM T60693 CRK2J6 73212901 EC50 = 0.41 nM T60693 CC65OA 73213195 Ki > 10000 nM T60693 CW83DK 73213196 Ki > 10000 nM T60693 COL97Y 73295685 IC50 = 12.6 nM T60693 CNA8O3 73345364 Ki = 3.39 nM T60693 CMU18J 73345366 Ki = 10 nM T60693 C7ZN1K 73345634 Ki = 28.18 nM T60693 CCN72S 73345747 IC50 = 12.75 nM T60693 CY03SQ 73346599 Ki = 1.28 nM T60693 CM0FA7 73346658 IC50 > 10000 nM T60693 CU7C6J 73346891 Ki = 0.44 nM T60693 C0T3UH 73347231 IC50 > 10000 nM T60693 CQJ36Z 73347341 EC50 = 0.077 nM T60693 CH2T1I 73347643 Ki = 136 nM T60693 C5HXL6 73347644 Ki = 4.05 nM T60693 C46QVZ 73348688 Ki = 30 nM T60693 CM70YA 73349151 Ki = 302 nM T60693 CW8A0Y 73349359 Ki = 1977 nM T60693 C5R1OC 73349360 Ki = 1662 nM T60693 C9Z3KC 73349647 Ki = 0.71 nM T60693 C0QE8Z 73350321 IC50 > 10000 nM T60693 CN5S4A 73350483 Ki = 681.3 nM T60693 C28LSE 73350518 Ki = 6.4 nM T60693 C5GAW0 73351393 EC50 = 3.8 nM T60693 C0W1NT 73351837 IC50 > 10000 nM T60693 CWA73N 73352217 Ki = 54 nM T60693 CL2W3H 73352233 Ki = 91 nM T60693 CSY9E4 73352234 EC50 = 5000 nM T60693 C7D1LF 73352661 Ki = 0.79 nM T60693 C3PZE0 73353313 IC50 > 10000 nM T60693 CKFA02 73353693 Ki = 39 nM T60693 C2NXP4 73354381 EC50 = 70 nM T60693 CO3ZS7 73354458 Ki = 1.2 nM T60693 COS31U 73354624 Ki = 282 nM T60693 C2HJ6O 73355223 Ki = 22 nM T60693 C4F7VK 73355415 Ki = 809 nM T60693 CAI63V 73355417 Ki = 4864 nM T60693 C3Z5LT 73355419 Ki = 934 nM T60693 C3Q9FB 73356023 Ki = 41.7 nM T60693 C83ZPI 73356767 Ki = 82 nM T60693 CJT8Y2 73356768 Ki = 198 nM T60693 C2E7QW 75201901 Ki = 3100 nM T60693 CSDY18 75441596 Ki = 6400 nM T60693 C1NQP6 76283714 Ki > 10000 nM T60693 CHJ1P9 76283716 Ki = 138.3 nM T60693 C81CHZ 76283968 Ki = 231.3 nM T60693 CC8U3Q 76283972 Ki = 1.86 nM T60693 CA4D6O 76284236 Ki = 0.94 nM T60693 C9PUY1 76308449 Ki = 7890 nM T60693 C89OES 76308450 Ki = 16000 nM T60693 C2LZD4 76309826 Ki = 0.14 nM T60693 CB78KL 76309827 Ki = 25.5 nM T60693 C68BLJ 76309828 Ki = 47.8 nM T60693 C35USC 76313542 Ki = 0.16 nM T60693 C6J2WF 76313543 Ki = 0.33 nM T60693 CZSU65 76313544 Ki = 0.26 nM T60693 C1GU9H 76317053 Ki = 148.2 nM T60693 CM9RC0 76317054 Ki = 0.12 nM T60693 CSYN97 76317055 Ki = 0.13 nM T60693 C0SWX7 76317056 Ki = 0.17 nM T60693 CP95SN 76317057 Ki = 67.2 nM T60693 CPKY85 76320762 Ki = 49.2 nM T60693 CG9MB3 76324401 Ki = 0.084 nM T60693 CU12ZJ 76324412 Ki = 7.79 nM T60693 CIX43W 76327982 Ki = 586.4 nM T60693 C6XT3U 76330188 Ki = 9910 nM T60693 CLU90M 76331610 EC50 = 0.61 nM T60693 CB4JI7 76331634 Ki = 46.6 nM T60693 CCW07O 76331635 Ki = 0.36 nM T60693 CRA1Y0 76331636 Ki = 0.33 nM T60693 C6F1BS 76335253 Ki = 0.27 nM T60693 COK40D 76335254 Ki = 0.19 nM T60693 CZP08R 76335255 Ki > 10000 nM T60693 C2LI9M 76440582 Ki = 6165.95 nM T60693 C3F2NW 77085815 Ki = 500 nM T60693 CLH3X9 81689704 Ki = 0.04 nM T60693 CTI5S8 81689720 Ki = 84.6 nM T60693 CGH7J9 86279209 Ki = 152 nM T60693 CD1OY5 86280667 EC50 = 2 nM T60693 C1WTJ6 86581710 EC50 = 2.2 nM T60693 CJ42SL 86648371 EC50 = 20 nM T60693 C5C9KE 86648372 EC50 = 150 nM T60693 CG1UD2 89001045 Ki = 10.3 nM T60693 C97GYK 89435126 Ki = 0.564 nM T60693 CL5R0T 89435196 EC50 = 0.2 nM T60693 C7X1VI 89435275 Ki = 2.43 nM T60693 C08YSC 89435280 Ki = 0.522 nM T60693 CZSC16 90306849 EC50 = 0.36 nM T60693 CR34DL 90306855 Ki = 0.16 nM T60693 C8HE3B 90306863 Ki = 0.39 nM T60693 C1W9QL 90306885 Ki = 2.8 nM T60693 CM5GS1 90306887 Ki = 0.1 nM T60693 C03HOW 90392373 Ki = 1.05 nM T60693 C0OAE4 90392376 Ki = 4.26 nM T60693 C47BLH 90397724 Ki = 0.362 nM T60693 C54EUB 90644257 Ki = 879 nM T60693 CZ10JE 90644258 Ki = 594 nM T60693 CV7U4P 90644259 Ki = 195 nM T60693 CI2TV6 90644873 Ki = 0.2 nM T60693 C3WD0A 90644874 Ki = 0.12 nM T60693 CGBL95 90644875 Ki = 0.08 nM T60693 C3VIY8 90645383 EC50 = 29 nM T60693 C18HBT 90645386 Ki = 9.4 nM T60693 C1DOG7 90654745 Ki > 375 nM T60693 CX3WT1 90654746 Ki > 375 nM T60693 CC70MH 90654747 Ki > 375 nM T60693 C4ZQD5 90654748 Ki > 375 nM T60693 CBV23K 90654749 Ki > 375 nM T60693 C87NYV 90654750 Ki > 375 nM T60693 C20FOK 90654751 Ki > 375 nM T60693 CT91LC 90654752 Ki > 375 nM T60693 CIQV28 90655825 EC50 = 333 nM T60693 C6V1PS 90655826 EC50 = 231 nM T60693 CNPC03 90655827 EC50 = 12530 nM T60693 CFAZ39 90655828 EC50 = 1.2 nM T60693 C63YPH 90655829 EC50 = 2.4 nM T60693 C7C5BM 90655970 Ki > 10000 nM T60693 CTV50C 90655971 Ki = 516 nM T60693 C1S5UB 90655972 Ki = 814 nM T60693 CV6A5T 90655973 Ki = 184 nM T60693 CL0D4Y 90655974 Ki = 56.3 nM T60693 C51CQN 90655975 Ki = 12.82 nM T60693 C2USA9 90655976 Ki = 88.4 nM T60693 CLKW80 90655977 Ki = 4171 nM T60693 C96DUE 90655978 Ki = 467.7 nM T60693 C1N5QA 90655979 Ki = 1367 nM T60693 C6FN2S 90656087 Ki = 134.9 nM T60693 C2QY3H 90656088 Ki = 25.2 nM T60693 CW2P5Q 90656089 Ki = 1.72 nM T60693 C8TV7C 90656090 EC50 > 5000 nM T60693 CK9FP8 90656664 Ki = 0.95 nM T60693 CC6LY3 90656665 EC50 = 2.1 nM T60693 COGW86 90656666 Ki = 0.56 nM T60693 C9YKV8 90656667 Ki = 0.75 nM T60693 C3WLH8 90656668 Ki = 0.36 nM T60693 CP1ZW6 90663949 Ki > 5000 nM T60693 CZ9GL5 90663950 Ki = 153 nM T60693 CFK27M 90663951 Ki = 779 nM T60693 CBT6F1 90663952 Ki > 5000 nM T60693 C1QAB3 90663953 Ki = 78 nM T60693 C5VZC6 90666479 Ki = 60 nM T60693 C2NG3A 90666726 Ki = 6.21 nM T60693 C5DG9V 90666727 Ki = 300 nM T60693 C26HUP 90666728 Ki = 75 nM T60693 CK0W6U 90666729 Ki = 81 nM T60693 CM75TG 90666730 Ki = 6.7 nM T60693 C4D6WT 90666731 Ki = 1233 nM T60693 C0GWK7 90666732 Ki = 5261 nM T60693 CT70RV 90666733 Ki = 7438 nM T60693 CT0O1B 90666734 Ki = 171 nM T60693 CCUK67 90666735 Ki = 462 nM T60693 CWI2S7 90666736 Ki = 59 nM T60693 C0BNE6 90667279 Ki = 142 nM T60693 CWOB91 90667280 Ki = 65 nM T60693 CU2XP8 91801212 EC50 = 9.95 nM T60693 CR93LZ 91928491 Ki > 10000 nM T60693 C2UZ4P 91928492 Ki > 10000 nM T60693 C1B6OP 92213238 EC50 = 2.2 nM T60693 CK4U6G 93967682 Ki = 1810 nM T60693 COM0Q7 94156776 Ki = 2690 nM T60693 CMI13V 95177310 Ki > 100000 nM T60693 CSPX47 95261164 Ki = 3140 nM T60693 C98WTN 95265878 Ki = 10500 nM T60693 C07VRA 101341769 Ki = 1900 nM T60693 CI4YM3 101806592 EC50 = 50.3 nM T60693 CW3LH2 101882818 Ki = 4.83 nM T60693 CW5H9D 101882819 Ki = 224 nM T60693 CGQV37 101882820 Ki = 1470 nM T60693 C5Z0DI 101886614 EC50 = 3.3 nM T60693 CNHS29 101898709 IC50 = 410 nM T60693 CJX06V 101910788 EC50 = 0.019 nM T60693 CO5Z0L 102014213 Ki = 2000 nM T60693 CPT9B3 102269996 Ki = 0.71 nM T60693 C9T1NI 102269998 Ki = 0.95 nM T60693 COFT20 102270003 Ki = 1.98 nM T60693 CR4KN5 102270004 Ki = 15.6 nM T60693 CP5F4Q 102270005 Ki = 182 nM T60693 C3FX4P 102270006 Ki = 4.68 nM T60693 CFA7K6 102270007 Ki = 48.7 nM T60693 CD19TA 102270008 Ki = 20.4 nM T60693 CTSL70 102497616 EC50 = 100 nM T60693 CH0KG6 117697800 EC50 = 1.2 nM T60693 C8P4XF 117705986 EC50 = 98 nM T60693 C0BCI6 117705988 EC50 = 404 nM T60693 CEP48V 117706009 Ki = 0.658 nM T60693 CMO27R 117706010 Ki = 1.38 nM T60693 C67SPE 117706054 EC50 = 0.3 nM T60693 C12FIV 117706085 Ki = 0.781 nM T60693 CIN6T1 117707041 EC50 = 8.1 nM T60693 CZ5AI6 117710394 EC50 = 1 nM T60693 C90PMZ 117710400 EC50 = 125 nM T60693 C3A7QZ 118200491 Ki = 2.7 nM T60693 CR52EZ 118200640 Ki = 4.6 nM T60693 CUCJ65 118263805 IC50 = 3 nM T60693 C9JV1T 118263857 IC50 = 7 nM T60693 CRY49P 118263892 IC50 = 1.3 nM T60693 C9YVS2 118263923 IC50 = 1.3 nM T60693 C5HCS3 118264001 IC50 = 2.2 nM T60693 C38LHY 118264112 IC50 = 1.3 nM T60693 CM8TB4 118705898 Ki = 0.15 nM T60693 C6RW0E 118705901 Ki = 0.33 nM T60693 C8ZM3D 118709349 Ki > 100000 nM T60693 C58BHC 118709350 Ki > 100000 nM T60693 C01ZSF 118709356 Ki > 100000 nM T60693 CK3S0G 118709357 Ki > 100000 nM T60693 CIJX58 118709358 Ki > 100000 nM T60693 CN3UC7 118709360 Ki > 100000 nM T60693 CW32LQ 118710801 EC50 = 64 nM T60693 CQ6O7Y 118710802 EC50 = 79 nM T60693 C27YCZ 118710804 EC50 = 470 nM T60693 CS9X1P 118710805 EC50 = 79 nM T60693 C0O5KT 118710807 EC50 = 170 nM T60693 CI1QT3 118711134 IC50 = 570 nM T60693 C4MRB0 118711135 IC50 = 370 nM T60693 CP6WQ1 118711209 IC50 = 1100 nM T60693 CL9F4B 118711887 Ki = 749 nM T60693 CBK60I 118713122 Ki = 18.1 nM T60693 C5J0UN 118713123 Ki = 385 nM T60693 CJ38GQ 118713124 Ki = 6 nM T60693 CCIS67 118713125 EC50 = 11 nM T60693 CDU9H7 118713126 Ki = 10 nM T60693 C8TPM0 118713127 Ki = 153 nM T60693 C9E8OS 118713128 Ki = 28.8 nM T60693 CRVW31 118713129 EC50 = 7 nM T60693 CO8UJ6 118713130 EC50 = 10 nM T60693 CL25HD 118713131 EC50 = 21 nM T60693 CI52KQ 118713132 EC50 = 38 nM T60693 C5MJX6 118713133 EC50 = 27 nM T60693 C4MHO8 118713134 EC50 = 1799 nM T60693 CT7EU4 118713135 EC50 = 50 nM T60693 CZFQ32 118713136 EC50 = 33 nM T60693 C0P3QL 118713137 EC50 = 32 nM T60693 CE4Z7B 118713138 EC50 = 20 nM T60693 C14HFW 118713139 EC50 = 642 nM T60693 C7HO5D 118713140 EC50 = 1210 nM T60693 C7NHP9 118713141 EC50 = 1762 nM T60693 CUY58S 118713142 Ki = 304 nM T60693 CQ7O8Y 118713832 EC50 = 2500 nM T60693 C8GHI5 118713833 EC50 > 10000 nM T60693 C5SA4Z 118713834 EC50 > 10000 nM T60693 C78LKO 118716009 EC50 = 0.033 nM T60693 C5BJA6 118716010 EC50 = 0.18 nM T60693 C5I8LR 118718683 Ki = 3.2 nM T60693 CV5IK0 118718684 Ki = 35.8 nM T60693 C79RZA 118718687 Ki = 83 nM T60693 C5LZB8 118718688 Ki = 60.1 nM T60693 C4E3IS 118718689 Ki > 10000 nM T60693 CAC2X3 118718690 Ki > 10000 nM T60693 C3CSD6 118718691 Ki = 75.7 nM T60693 CIUQ43 118718718 Ki > 10000 nM T60693 CU10SI 118722557 Ki = 159 nM T60693 CTNV42 118723390 EC50 = 8.4 nM T60693 CP2IQ1 118723391 EC50 = 27 nM T60693 C6LV7N 118723392 EC50 = 1020 nM T60693 C28MTF 118723393 EC50 = 1.2 nM T60693 CG5ER8 118723394 EC50 = 12 nM T60693 CXM3E1 118723395 EC50 = 54 nM T60693 C92XIR 118723396 EC50 = 360 nM T60693 CZTJ31 118723397 EC50 = 450 nM T60693 COSU53 118723398 EC50 = 170 nM T60693 CDIQ78 118723399 EC50 = 5.4 nM T60693 CBTD92 118723400 EC50 = 3.4 nM T60693 C5Z4UM 118723401 EC50 = 2.3 nM T60693 CEK87Z 118723402 EC50 = 10 nM T60693 CIBL50 118723403 EC50 = 8.6 nM T60693 C9D7ZO 118723404 EC50 = 37 nM T60693 C9SL2Y 118723405 EC50 = 25 nM T60693 C7WT5D 118723840 EC50 = 6.5 nM T60693 CP2XB1 118723841 EC50 = 4.3 nM T60693 CQ72AL 118723842 EC50 = 1 nM T60693 C0JMR8 118723843 EC50 = 20 nM T60693 CWG9H5 118723844 EC50 = 38 nM T60693 C4M1EP 118723845 EC50 = 26 nM T60693 CT0C1O 118723846 EC50 = 6100 nM T60693 CB32DY 118723847 EC50 = 430 nM T60693 C8S5TQ 118723848 EC50 = 9250 nM T60693 C59ZOP 118723849 EC50 = 890 nM T60693 C8G7RP 118723850 EC50 = 2.9 nM T60693 CB1J4T 118723851 EC50 = 430 nM T60693 C8KHZ6 118723852 EC50 = 630 nM T60693 CVE6B7 118723853 EC50 = 620 nM T60693 C8TNG6 118723854 EC50 = 240 nM T60693 CL1ID4 118723855 EC50 = 250 nM T60693 CFI53Q 118723856 EC50 = 3.1 nM T60693 CS5Y2A 118723857 EC50 = 31 nM T60693 CF81XL 118723858 EC50 = 7.3 nM T60693 C0ZE4P 118723859 EC50 = 9.4 nM T60693 CA51CQ 118724536 Ki > 5000 nM T60693 CH4LB0 118724977 Ki = 1233 nM T60693 C9SN0M 118724979 Ki = 705 nM T60693 CH9GT5 118724980 Ki = 3678 nM T60693 CG7SQ8 118724984 Ki = 4247 nM T60693 C7L6ZT 118725739 EC50 = 878 nM T60693 C06YTM 118725740 EC50 = 1400 nM T60693 C29CVM 118725741 EC50 = 33 nM T60693 C1GE2L 118725742 EC50 = 423 nM T60693 C8VDF6 118725743 EC50 = 355 nM T60693 C1U9MH 118725744 EC50 = 1225 nM T60693 C0HM6Y 118725745 EC50 = 72 nM T60693 C4NV9S 118725746 EC50 = 1550 nM T60693 C10UTX 118725747 EC50 = 4250 nM T60693 CW70QU 118725748 EC50 > 10000 nM T60693 C0CJT4 118725749 EC50 > 10000 nM T60693 CW9NF2 118725750 EC50 = 537 nM T60693 CDC3J4 118725751 EC50 = 970 nM T60693 CI1CY5 118725752 EC50 = 478 nM T60693 C2M6JZ 118725753 EC50 > 10000 nM T60693 CDLN25 118725754 EC50 = 118 nM T60693 C6FLS7 118725836 EC50 = 2950 nM T60693 C9CG6P 118725837 EC50 = 2400 nM T60693 C1ZB3U 118725838 EC50 = 10000 nM T60693 CG4UH3 118725839 EC50 = 1550 nM T60693 CT61VY 118725840 EC50 = 1800 nM T60693 CXL16I 118725841 EC50 = 7 nM T60693 COA5Z4 118725842 EC50 = 2050 nM T60693 C49YCX 118725843 EC50 = 70 nM T60693 CSB20M 118725844 EC50 = 152 nM T60693 CBU3D5 118725845 EC50 = 1050 nM T60693 CU8VY6 118725846 EC50 = 734 nM T60693 CX4E9W 118725847 EC50 > 10000 nM T60693 CCQ85P 118725848 EC50 = 22 nM T60693 C1Q5IB 118725849 EC50 = 122 nM T60693 CE86DJ 118725850 EC50 = 8 nM T60693 C2YR9E 118725851 EC50 = 1440 nM T60693 CVC2R9 118725852 EC50 = 765 nM T60693 CBDA90 118725853 EC50 = 1 nM T60693 CET5Y3 118725854 EC50 = 31 nM T60693 C2LA6F 118725855 EC50 = 2 nM T60693 CO8B9L 118725856 EC50 = 10 nM T60693 CMO86W 118725857 EC50 = 37 nM T60693 C61VHK 118725858 EC50 = 395 nM T60693 C1UD6R 118726271 IC50 = 200 nM T60693 CQH1G3 118731120 Ki = 29.9 nM T60693 CDN86Z 118731405 Ki = 110 nM T60693 CK5W7M 118731406 Ki = 110 nM T60693 C29ESD 118731407 Ki = 160 nM T60693 CAP48T 118731408 Ki = 88 nM T60693 C12NJU 118731409 Ki = 139 nM T60693 CM06BI 118731410 Ki = 5.1 nM T60693 CP84KM 118731411 Ki = 1.4 nM T60693 C5MK1D 118731412 Ki = 795 nM T60693 CPD5R9 118731413 Ki = 923 nM T60693 CY9NH0 118731414 Ki = 117 nM T60693 CR6K5D 118731415 Ki = 147 nM T60693 CMR93J 118731416 Ki = 230 nM T60693 CQ39OA 118731417 Ki = 424 nM T60693 CK76UL 118731418 Ki = 163 nM T60693 CRXY76 118731419 Ki = 1.6 nM T60693 C9A4RX 118731420 Ki = 1769 nM T60693 CC2S7I 118731421 Ki = 410 nM T60693 C3N0VC 118731422 Ki = 3184 nM T60693 C4FT8K 118731423 Ki = 82 nM T60693 C1L4QH 118731424 Ki = 130 nM T60693 CB0R9K 118731425 Ki = 177 nM T60693 CW35DR 118731426 Ki = 297 nM T60693 CP61XB 118731427 Ki = 3.7 nM T60693 CD51ZQ 118731428 Ki = 1119 nM T60693 C14DLY 118872292 EC50 = 4000 nM T60693 CTC59H 121308699 EC50 = 351 nM T60693 CWO42N 121365644 IC50 = 1.6 nM T60693 C3E1HM 121365654 IC50 = 10 nM T60693 CG52CR 121365655 IC50 = 19.7 nM T60693 C3L8IJ 121365661 IC50 = 930 nM T60693 CI57VQ 121365662 IC50 = 33 nM T60693 CWSZ03 121373658 IC50 = 3.7 nM T60693 CG6X8L 121373661 IC50 = 87 nM T60693 C6DBM3 121373662 IC50 = 85 nM T60693 CBTJ31 121373663 IC50 = 106 nM T60693 CAHC31 121373668 IC50 = 29.1 nM T60693 CTZ5D3 121373677 IC50 = 143 nM T60693 C9ND2K 121373679 IC50 = 5.3 nM T60693 CP1D8B 121614426 IC50 = 140 nM T60693 CSRW32 121614490 IC50 = 8930 nM T60693 C6KIU4 121614638 IC50 = 260 nM T60693 CC3E1H 121614661 IC50 = 50 nM T60693 CQ3LD2 121614853 IC50 = 570 nM T60693 CWP9E2 122178420 EC50 = 4.898 nM T60693 CQ7YP3 122178421 EC50 = 11.75 nM T60693 C5QZT2 122178422 EC50 = 4.786 nM T60693 C74MRY 122178423 EC50 = 2.818 nM T60693 C5JCY2 122178425 EC50 = 2.239 nM T60693 C1A2JB 122178426 EC50 = 1.349 nM T60693 CMH98S 122178427 EC50 = 3.631 nM T60693 CK0LH7 122179050 Ki = 0.08 nM T60693 CBP42W 122179052 Ki = 0.04 nM T60693 CNCJ68 122179053 Ki = 0.05 nM T60693 CY96XI 122179055 Ki = 0.12 nM T60693 C6LDU5 122179056 Ki = 0.11 nM T60693 C57GMN 122179057 Ki = 0.16 nM T60693 C0X6AF 122179058 Ki = 0.1 nM T60693 C09BYL 122179060 Ki = 0.094 nM T60693 CF83LN 122179061 Ki = 0.13 nM T60693 C6YQM4 122179064 Ki = 0.14 nM T60693 CRKB15 122179557 EC50 = 10 nM T60693 C8OF5S 122179558 EC50 = 7.586 nM T60693 C0WKQ3 122179559 EC50 = 72.44 nM T60693 C93YZC 122179560 EC50 = 1.047 nM T60693 CZ6KB3 122181405 IC50 > 18000 nM T60693 C3UV6A 122182776 Ki = 468 nM T60693 CVMP98 122182777 Ki = 74.3 nM T60693 C20HCF 122182778 Ki = 397 nM T60693 C3S5RY 122182780 Ki > 1000 nM T60693 C18PTI 122182782 Ki > 1000 nM T60693 C6R8UI 122182784 Ki = 477 nM T60693 CG7N6Q 122182786 Ki = 313 nM T60693 CYJ34R 122182788 Ki = 854 nM T60693 CDJ0N9 122182790 Ki > 1000 nM T60693 CWYQ85 122182792 Ki > 1000 nM T60693 C80PUY 122183206 Ki = 200 nM T60693 C61ZWM 122183207 Ki = 340 nM T60693 CP7G1A 122183208 Ki = 45 nM T60693 C6GLF5 122183209 Ki = 100 nM T60693 CIP5Y3 122183210 Ki = 19 nM T60693 C9YU5A 122183211 Ki = 59 nM T60693 CIL5O7 122183212 Ki = 430 nM T60693 CMR9Q4 122183213 Ki = 11 nM T60693 CULZ39 122183217 Ki = 340 nM T60693 C0CPO2 122183218 Ki = 42 nM T60693 CDUW32 122183219 Ki = 2.3 nM T60693 CA7R3L 122183220 Ki = 14 nM T60693 C7EO2T 122183221 Ki = 9.7 nM T60693 C7QKU8 122183222 Ki = 78 nM T60693 CA0B9X 122183223 Ki = 39 nM T60693 CXE52Q 122183281 Ki = 71 nM T60693 CV0FU5 122183282 Ki = 11 nM T60693 CEP3K5 122183283 Ki = 52 nM T60693 CB9Z1T 122183284 Ki = 12 nM T60693 C27DRW 122188793 EC50 = 11.8 nM T60693 C9IDJ8 122191987 Ki > 1000 nM T60693 CMH0N5 122191988 Ki > 1000 nM T60693 CX26TV 122191989 Ki = 210 nM T60693 C02ACR 122191990 Ki = 301 nM T60693 CV5QH9 122191991 Ki = 20.5 nM T60693 C6MG0O 122191992 Ki = 4.7 nM T60693 CM0F3R 122191993 Ki = 48 nM T60693 C8TZ0N 122191994 Ki = 250 nM T60693 CY8P6A 122191995 Ki > 1000 nM T60693 CNW0S1 122191996 Ki > 1000 nM T60693 C03RUP 122191997 Ki = 108 nM T60693 CNL14S 122191998 Ki = 316 nM T60693 CNE13U 122194668 Ki = 28.6 nM T60693 C50YUK 122195953 Ki = 87 nM T60693 CXD3P2 122195954 Ki = 19 nM T60693 CUX4S3 122195955 Ki = 6.2 nM T60693 CZT35A 122195956 Ki = 8.4 nM T60693 CA8JB7 122195957 Ki = 20 nM T60693 C1FC5Z 122195958 Ki = 48 nM T60693 CW17NE 122195959 Ki = 92 nM T60693 CE7BZ0 122195960 Ki = 4.3 nM T60693 CHU84Z 122195961 Ki = 63 nM T60693 CT8X2B 122195962 Ki = 12 nM T60693 CU4CT0 122195963 Ki = 19 nM T60693 CA9O5R 122195964 Ki = 15 nM T60693 CCQ3E0 122197314 IC50 > 10000 nM T60693 C5K8XH 122197315 IC50 > 10000 nM T60693 CFWE98 122197316 IC50 > 9960 nM T60693 CZ03XS 122197485 IC50 = 7200 nM T60693 C0WTE6 122197486 IC50 = 7000 nM T60693 C1TP0H 122197487 IC50 > 6000 nM T60693 CSN3V4 122197488 IC50 > 6400 nM T60693 C6LC2J 122197489 IC50 > 5800 nM T60693 CPCF21 122197490 IC50 = 2020 nM T60693 CF8X5R 122197491 IC50 > 9500 nM T60693 CMA83V 122197492 IC50 = 204 nM T60693 CX4I7N 122197493 IC50 = 961 nM T60693 CWZA97 122197494 IC50 > 10000 nM T60693 CTKY87 122197495 IC50 > 4900 nM T60693 CH9O2Q 122197496 IC50 = 6920 nM T60693 C5I8CM 122197497 IC50 = 6100 nM T60693 C7EF4P 122197498 IC50 = 1600 nM T60693 C1BDZ4 122197499 IC50 = 31 nM T60693 C7F8CK 122197500 IC50 > 10000 nM T60693 CMH7K2 122197501 IC50 > 10000 nM T60693 CD3L6S 122197502 IC50 > 10000 nM T60693 C7O1EP 122197503 IC50 > 10000 nM T60693 CYE18M 122197504 IC50 = 3200 nM T60693 C9W2FQ 122197505 IC50 = 3600 nM T60693 C45VUL 122197506 IC50 > 10000 nM T60693 CEP3J0 122197507 IC50 = 7400 nM T60693 C9B5DC 122197508 IC50 > 10000 nM T60693 CZTO90 122197509 IC50 > 4000 nM T60693 C7SJO2 122197510 IC50 > 75000 nM T60693 CH93LB 122197511 IC50 = 5330 nM T60693 CL78AV 122197512 IC50 = 1200 nM T60693 CAQ5B0 122409965 Ki = 732 nM T60693 C0K8BS 122589938 Ki = 79.1 nM T60693 CBU38O 122589952 Ki = 36.3 nM T60693 CTNU73 123445395 Ki = 7500 nM T60693 C9FBD2 127025219 Ki = 1.3 nM T60693 CL3VG1 127025528 Ki = 0.18 nM T60693 C5D7WM 127025817 Ki = 0.049 nM T60693 CTBN56 127026052 Ki = 2187.76 nM T60693 CKP92G 127026454 EC50 = 1288.25 nM T60693 CI3YF5 127026455 EC50 = 1698.24 nM T60693 CRDW90 127026456 EC50 = 41.69 nM T60693 CO5S0Z 127026457 EC50 = 102.33 nM T60693 C7IF4H 127028132 Ki = 130 nM T60693 CUEQ87 127028133 Ki = 2500 nM T60693 CFR0V8 127028436 EC50 = 370 nM T60693 CP0YZ3 127028437 Ki = 35 nM T60693 CUQJ15 127029584 Ki = 96 nM T60693 CSK04O 127032208 EC50 = 3.19 nM T60693 CR3TB5 127032209 Ki = 3.22 nM T60693 C2SP1T 127032210 Ki = 4.3 nM T60693 CXJY65 127032211 EC50 = 8.02 nM T60693 CK29CG 127032212 Ki = 9.11 nM T60693 CQ25BG 127032213 Ki = 9.65 nM T60693 CY72AX 127033106 Ki = 31 nM T60693 CN0BZ9 127033398 Ki = 0.748 nM T60693 CFR46S 127033399 Ki = 2.97 nM T60693 CML91J 127033967 Ki = 17.5 nM T60693 CZ61LK 127034966 EC50 > 5011.87 nM T60693 CA0SN5 127034967 EC50 > 5011.87 nM T60693 CQ0ZT9 127035062 Ki = 363 nM T60693 CU49VE 127036186 Ki = 1230.27 nM T60693 CG06BD 127036932 Ki = 812.83 nM T60693 CVW71O 127036953 Ki = 891.25 nM T60693 CYN01M 127041368 EC50 = 812.83 nM T60693 CXMJ48 127043001 Ki = 84 nM T60693 CM6RV9 127043037 Ki = 3.56 nM T60693 CEGF25 127043063 Ki > 10000 nM T60693 C0CMH9 127043073 Ki > 10000 nM T60693 C3W5SX 127043074 Ki > 10000 nM T60693 CQVP14 127043075 Ki > 10000 nM T60693 C32KON 127043249 Ki > 10000 nM T60693 C7CKP3 127043256 Ki > 10000 nM T60693 C7XF0S 127043262 Ki > 10000 nM T60693 C4LOH0 127043264 Ki = 140 nM T60693 CL25KU 127043277 Ki > 10000 nM T60693 CFU4H9 127043364 Ki = 47 nM T60693 CUX47D 127043424 Ki > 10000 nM T60693 CCP2Z8 127043425 Ki > 10000 nM T60693 C7HM0D 127043432 Ki > 10000 nM T60693 C0WM8J 127043433 Ki > 10000 nM T60693 C8CV6X 127043434 Ki > 10000 nM T60693 C30BNK 127043559 Ki = 22 nM T60693 C1GK3A 127043614 Ki > 10000 nM T60693 C61FHR 127043615 Ki > 10000 nM T60693 CCSZ68 127044528 Ki = 33 nM T60693 C71EWR 127045653 Ki = 1540 nM T60693 CE1A7K 127045654 Ki = 4400 nM T60693 CTA96D 127045655 Ki = 230 nM T60693 C61KVS 127046953 Ki = 800 nM T60693 C83YWS 127046954 Ki = 2900 nM T60693 CZ3CY2 127046955 Ki = 6470 nM T60693 CPR6J4 127049272 Ki = 25 nM T60693 CD5XV4 127049273 Ki = 56 nM T60693 CAN7H2 127049274 Ki = 29 nM T60693 CLRT48 127049275 Ki = 34 nM T60693 C85ZFT 127049276 Ki = 39 nM T60693 C9VFJ2 127050108 Ki = 40 nM T60693 CLB51H 127050830 Ki = 4.3 nM T60693 C6ZGX7 127050831 Ki = 15 nM T60693 CIB0Z8 127050832 Ki = 280 nM T60693 CNS8M3 127050833 Ki = 58 nM T60693 CIBX04 127050834 Ki = 64 nM T60693 CM8O4S 127051732 Ki = 50 nM T60693 C5BU6I 127051733 Ki = 76 nM T60693 CSN5R2 127053153 Ki = 190 nM T60693 C4SU9L 129093829 Ki > 1000 nM T60693 C1EHU5 129188443 Ki = 1594 nM T60693 CD8FT9 129188454 Ki > 10000 nM T60693 CC9Z0J 129188459 Ki = 562 nM T60693 C50GOC 130442480 Ki = 7200 nM T60693 CM04RF 130442572 Ki = 1500 nM T60693 C1RI8Q 132060720 Ki = 3182 nM T60693 CWQO32 132584396 Ki > 10000 nM T60693 CENF10 132584397 Ki = 3624 nM T60693 CM1PN3 132584398 Ki = 1695 nM T60693 CS2H6B 132584403 Ki > 10000 nM T60693 CAVB41 132584404 Ki = 416 nM T60693 CO69MW 134130798 Ki = 1602 nM T60693 CA1V9U 134131635 Ki > 10000 nM T60693 C4GPT2 134131885 Ki = 1396 nM T60693 C3Z6SV 134131949 Ki > 10000 nM T60693 C64JNH 134134355 Ki > 10000 nM T60693 C91TWF 134134844 Ki > 10000 nM T60693 C7A1PO 134137537 Ki = 278 nM T60693 CL4K1Z 134139120 Ki > 10000 nM T60693 CK2X3O 134139232 Ki = 1276 nM T60693 C80ZPT 134139387 Ki = 211 nM T60693 CSX32C 134141708 Ki > 10000 nM T60693 CC8V6M 134142063 Ki > 10000 nM T60693 CTQ91W 134142390 Ki > 10000 nM T60693 CG0V4O 134142896 Ki > 10000 nM T60693 CBG64F 134144504 Ki = 3488 nM T60693 CU3L0J 134145684 Ki = 1229 nM T60693 CGV52O 134147031 Ki = 218 nM T60693 C5VAD3 134147144 Ki > 10000 nM T60693 C62SOQ 134147564 Ki = 711 nM T60693 C8DP6W 134147710 Ki = 372 nM T60693 CB8CI0 134147910 Ki = 1474 nM T60693 CBU81N 134149168 Ki > 10000 nM T60693 C5ZD9L 134149737 Ki > 10000 nM T60693 CH97MA 134154487 Ki = 493 nM T60693 CT2X3N 134155538 Ki > 10000 nM T60693 C9QBY4 134156534 Ki > 10000 nM T60693 C13PHC 134157413 Ki = 638 nM T60693 CLS5H3 134227139 Ki = 0.6 nM T60693 CG57MT 134563466 Ki = 1328 nM T60693 CE5RS7 134563496 Ki > 10000 nM T60693 CAEY19 134563500 Ki = 3456 nM T60693 C82SEF 134563650 Ki > 10000 nM T60693 CC3HK6 134563655 Ki = 172 nM T60693 C4U9EM 134563691 Ki > 10000 nM T60693 CFX37T 134563695 Ki = 446 nM T60693 CPEH72 134563698 Ki = 81 nM T60693 CR74XA 134563699 Ki = 830 nM T60693 C9PN6I 134578342 Ki = 1440 nM T60693 CK62WY 134578456 Ki > 10000 nM T60693 CN0C9Z 134578457 Ki = 461 nM T60693 C0HNI9 134578506 Ki = 3840 nM T60693 C0JCQ2 134578518 Ki = 1490 nM T60693 C1GY2T 135156251 EC50 > 10000 nM T60693 CPZ89B 135314564 Ki > 1000 nM T60693 CAX4E7 135329044 IC50 = 2.3 nM T60693 CG7P3W 135329090 IC50 = 2.4 nM T60693 CMS56H 135329094 IC50 = 2.1 nM T60693 CUYV98 135329104 IC50 = 3.6 nM T60693 CRW47P 135329122 IC50 = 4.5 nM T60693 CO87XZ 135445735 Ki = 0.0048 nM T60693 CP67DS 136112814 Ki = 8100 nM T60693 CWE6O8 136126655 Ki = 12 nM T60693 C8IP5C 136126656 Ki = 160 nM T60693 C7FW4R 136239492 Ki > 10000 nM T60693 CC6OP7 136244089 Ki > 10000 nM T60693 CQKN40 137434120 IC50 = 0.53 nM T60693 C0PL4B 137434175 IC50 = 0.8 nM T60693 CNCS34 137434196 IC50 = 0.78 nM T60693 CW8LH6 137434204 IC50 = 1.1 nM T60693 COQ5H7 137434366 IC50 = 0.88 nM T60693 C2JK8N 137434496 IC50 = 0.26 nM T60693 CX2N7C 137541775 IC50 = 140 nM T60693 CF4UH6 137541784 IC50 = 440 nM T60693 C2O3XI 137541786 IC50 = 810 nM T60693 C8H2LE 137541793 IC50 = 2940 nM T60693 CVBP38 137541794 IC50 = 90 nM T60693 C0OKP7 137541796 IC50 = 780 nM T60693 C3QB8I 137541808 IC50 = 1120 nM T60693 C07WHM 137541810 IC50 = 80 nM T60693 CW6SK2 137541816 IC50 = 490 nM T60693 C48SIG 137628671 Ki = 2290 nM T60693 C0BKU3 137631438 Ki = 4603 nM T60693 CD6OS8 137631684 EC50 = 0.028 nM T60693 CTH8M9 137631847 Ki = 0.14 nM T60693 CIW57H 137631944 IC50 = 910 nM T60693 CRYL80 137632074 EC50 = 1.7 nM T60693 C9WUL6 137632260 Ki > 1000 nM T60693 CNC15K 137632903 Ki = 3.56 nM T60693 C6FEL8 137633728 Ki = 3.99 nM T60693 CPG3W6 137633864 EC50 = 1.4 nM T60693 CY7KF5 137634296 EC50 = 8 nM T60693 CBW57P 137634403 Ki = 0.71 nM T60693 CB14RN 137635022 Ki = 176 nM T60693 C4LA6R 137635412 EC50 = 5.9 nM T60693 C9WI8Z 137635660 IC50 = 1800 nM T60693 C4UD2N 137636954 EC50 = 5 nM T60693 CIT2D7 137637157 EC50 = 0.3 nM T60693 CXB49H 137637261 EC50 = 5.04 nM T60693 C5EO6T 137637552 Ki = 42.7 nM T60693 CTQ24N 137637610 EC50 = 0.4 nM T60693 CUG84V 137637659 EC50 = 0.0257 nM T60693 C7I1NR 137638013 EC50 = 2.2 nM T60693 C3NT7A 137638511 Ki = 70.4 nM T60693 C6IE4A 137638534 EC50 > 100 nM T60693 CKR9S7 137638688 Ki = 0.017 nM T60693 C8JHP6 137638874 Ki = 31 nM T60693 CH4RQ3 137639037 EC50 = 0.0799 nM T60693 C4A7CD 137639500 EC50 = 7.51 nM T60693 C4CWP3 137639680 Ki = 29.4 nM T60693 CN25HL 137639933 EC50 = 0.9 nM T60693 C2LAX8 137639991 EC50 = 11 nM T60693 C9A2VZ 137640408 Ki = 3000 nM T60693 CL8KE4 137640513 EC50 = 2.2 nM T60693 CX7N6Q 137640628 EC50 = 1.8 nM T60693 CUZ7O1 137640860 Ki = 2.1 nM T60693 CY2AV8 137641064 Ki = 793 nM T60693 C2OD0K 137641318 Ki > 1000 nM T60693 CMI3T0 137641479 IC50 = 9.32 nM T60693 CF7Q8M 137641618 Ki = 7.92 nM T60693 C1RAK0 137642012 Ki = 0.31 nM T60693 CC7HE1 137642394 EC50 = 14 nM T60693 C1IAZ5 137642772 Ki = 209 nM T60693 C8BZ5G 137642854 EC50 = 0.0494 nM T60693 C4KT5V 137642888 EC50 = 0.291 nM T60693 CQ9NY2 137642933 EC50 = 0.00466 nM T60693 CKH93R 137643506 Ki = 0.072 nM T60693 CAI9Z4 137643649 Ki = 1738 nM T60693 CE0N8Y 137643858 EC50 > 10000 nM T60693 CU7MG5 137644005 Ki > 1000 nM T60693 C2MRK0 137645329 Ki > 1000 nM T60693 C21WKZ 137645421 EC50 = 4.5 nM T60693 C91QRT 137646062 EC50 = 3.9 nM T60693 CG4N0O 137646080 Ki = 1067 nM T60693 CUHF67 137646492 EC50 = 0.0222 nM T60693 C2OB5H 137646522 Ki = 0.12 nM T60693 CB34GJ 137646619 EC50 = 0.0288 nM T60693 CXJ9G7 137646782 Ki = 1.85 nM T60693 C3MV2Q 137646937 Ki = 37.6 nM T60693 CEO40K 137647271 EC50 = 1.5 nM T60693 CO7CV8 137647517 IC50 = 1400 nM T60693 CTP82Z 137647554 Ki = 10.3 nM T60693 CU36EQ 137647949 EC50 = 0.6 nM T60693 CX72UG 137648224 Ki = 5461 nM T60693 CK8EP7 137648628 Ki = 884 nM T60693 CH8F7A 137649449 Ki = 6717 nM T60693 C8M6VC 137649460 EC50 = 30 nM T60693 C4TDX9 137649850 Ki = 2.69 nM T60693 CH84NE 137651461 EC50 = 0.0283 nM T60693 CZ68WR 137651510 Ki = 19.1 nM T60693 C2P9ZA 137652088 EC50 > 10000 nM T60693 CK74TN 137652971 Ki = 126 nM T60693 C9YHQ5 137653349 Ki = 4625 nM T60693 C49ZTG 137653556 EC50 = 15 nM T60693 CS1B3U 137654001 Ki = 3.37 nM T60693 CL80PT 137654768 EC50 = 13 nM T60693 C9HWV3 137654943 EC50 = 11.7 nM T60693 C6N8JM 137655206 Ki = 3.43 nM T60693 C7P9UA 137655599 Ki = 0.061 nM T60693 C3KPA4 137655663 Ki = 602 nM T60693 CQR50I 137656159 EC50 = 6.9 nM T60693 C7Y5PH 137656268 EC50 = 8.1 nM T60693 C4D8UC 137656339 EC50 = 0.122 nM T60693 CAB49D 137656834 EC50 > 10000 nM T60693 CSHN48 137656887 Ki = 4.62 nM T60693 CY21WB 137657032 Ki = 0.221 nM T60693 C9QLZ8 137657690 EC50 = 761 nM T60693 CWD31I 137657725 Ki = 0.85 nM T60693 C9CJL2 137657927 IC50 = 1862.09 nM T60693 C2OK6H 137658170 EC50 = 4.7 nM T60693 CY94PV 137658980 IC50 = 800 nM T60693 CVU76G 137659256 EC50 > 100 nM T60693 CM85RN 137659520 EC50 = 1.04 nM T60693 C0K9SV 137659967 EC50 = 0.0953 nM T60693 CG8R9U 137660781 Ki = 0.04 nM T60693 CR0EW1 137660824 Ki = 0.38 nM T60693 C1XPN8 137661045 Ki = 200 nM T60693 C50LAS 137661659 EC50 = 3.2 nM T60693 CNX2Q5 137662177 Ki > 1000 nM T60693 C9LM6E 137662178 Ki = 43.5 nM T60693 CDA24L 145950961 Ki > 100000 nM T60693 C7WT1M 145952813 Ki > 100000 nM T60693 C7SX5C 145957352 IC50 = 0.22 nM T60693 C7X0LW 145958562 Ki > 100000 nM T60693 CY1MB9 145961131 Ki = 5.6 nM T60693 CR8WC1 145961165 Ki = 17.38 nM T60693 CIU2V6 145961844 Ki = 0.87 nM T60693 CGR0Y1 145963106 Ki = 18.62 nM T60693 CBFE94 145963594 Ki = 4.898 nM T60693 CL9M7U 145964011 Ki = 5.3 nM T60693 CH0VD5 145964426 Ki = 720 nM T60693 C85HUP 145965612 EC50 = 16000 nM T60693 CFW12R 145965818 Ki = 35 nM T60693 C0ZA3K 145965848 EC50 = 8000 nM T60693 CCYN90 145966041 EC50 > 50000 nM T60693 CUM96J 145966903 EC50 = 6000 nM T60693 CX64CN 145967261 EC50 > 50000 nM T60693 CR34HG 145969839 Ki = 179 nM T60693 CZ3NW6 145971020 EC50 > 50000 nM T60693 C47YPS 145972508 EC50 = 2000 nM T60693 CT5CX0 145973771 Ki = 4060 nM T60693 CKQY21 145974323 Ki = 4670 nM T60693 CAUE51 145974936 Ki = 6.7 nM T60693 C6EX7P 145977620 EC50 = 12000 nM T60693 CQS9N0 145978012 Ki = 6.7 nM T60693 C87MSW 145980271 Ki = 10000 nM T60693 C8I7QL 145980875 Ki = 1705 nM T60693 C63FHK 145982510 Ki = 48.5 nM T60693 C36TEU 145982515 Ki = 168.8 nM T60693 CC6A9H 145982585 Ki = 11.3 nM T60693 CU2IK5 145982792 Ki = 1250 nM T60693 CTQV67 145982828 EC50 = 87.2 nM T60693 C8MY6V 145982968 Ki = 38 nM T60693 CO8Z4U 145983526 Ki = 2.1 nM T60693 C4L7PT 145983969 Ki = 9.1 nM T60693 CK6F1J 145984022 Ki = 303.2 nM T60693 C1ONP2 145984192 Ki = 28 nM T60693 COP2I9 145984332 Ki = 0.4 nM T60693 C4KS7H 145984702 Ki = 33.2 nM T60693 CTY73C 145984984 Ki = 9 nM T60693 CW3H4T 145986047 EC50 = 3.3 nM T60693 C4N3JP 145986165 Ki = 72.1 nM T60693 CNJH37 145986752 Ki = 10000 nM T60693 CUGO10 145988693 Ki = 667 nM T60693 C0FT8Y 145991902 Ki = 0.17 nM T60693 CCP2U1 145992489 Ki = 1021 nM T60693 CW42UE 145993745 Ki = 30 nM T60693 C2ADQ5 145994326 EC50 = 492.4 nM T60693 C3CP1R 145994327 EC50 > 1000 nM T60693 CFO47R 145994330 EC50 > 1000 nM T60693 CBFX85 145994331 EC50 > 1000 nM T60693 CF7GX6 145994332 EC50 > 1000 nM T60693 CL69BD 145994333 EC50 > 1000 nM T60693 CSE72Q 145994334 EC50 > 1000 nM T60693 CW6I7K 145994336 EC50 > 1000 nM T60693 C0YWU3 145994337 EC50 > 1000 nM T60693 CVK19A 145994338 EC50 > 1000 nM T60693 CT3MY4 145994339 EC50 > 1000 nM T60693 C23IEG 145994341 EC50 > 1000 nM T60693 CZC6W1 145994342 EC50 = 134.8 nM T60693 C9RJO2 145994343 EC50 = 26.79 nM T60693 CG9XC0 145994345 EC50 = 258.2 nM T60693 CC2G1V 146025727 Ki = 3200 nM T60693 C6P3SR 153287553 Ki > 10000 nM T60693 CV9G7Z 153287572 Ki > 10000 nM T60693 CO85KL 153287574 Ki > 10000 nM T60693 CL6OY2 155510745 Ki = 495 nM T60693 CA3MB9 155511121 EC50 = 75.5 nM T60693 CY8GO4 155511793 Ki = 16.1 nM T60693 C4H6VE 155511829 Ki = 370 nM T60693 CQ58SJ 155512448 Ki = 528 nM T60693 CVMK78 155512747 Ki = 247 nM T60693 CG95UQ 155512955 Ki = 1.1 nM T60693 C0AW7D 155513170 EC50 = 32 nM T60693 C8AJS3 155513639 Ki = 16.9 nM T60693 CT19NM 155514601 Ki = 408 nM T60693 C1UXA4 155514661 Ki = 44.2 nM T60693 CKL4N0 155515090 IC50 = 9.5 nM T60693 CUM2N4 155515982 Ki = 3900 nM T60693 C7RT4P 155516535 Ki = 261 nM T60693 C3MQP5 155516545 Ki > 716 nM T60693 C8U0GP 155516761 Ki = 49.5 nM T60693 C3PD8O 155516811 Ki = 243 nM T60693 CJ80FA 155516945 IC50 = 10.3 nM T60693 CN0KZ4 155517081 Ki = 68 nM T60693 C6VP0Q 155517279 Ki = 1588 nM T60693 CUD1L3 155518099 Ki = 116 nM T60693 C5HXW8 155518735 Ki > 100000 nM T60693 C7ZO4J 155518809 Ki = 40.3 nM T60693 C3RU8T 155518842 Ki = 117 nM T60693 C5SE3P 155519089 Ki = 17.2 nM T60693 CL7C8R 155519639 Ki = 319 nM T60693 CUSA24 155519891 Ki > 10000 nM T60693 CRKM35 155520586 Ki = 0.47 nM T60693 CU4K8P 155521065 Ki = 16.8 nM T60693 CR80YQ 155521541 Ki = 330 nM T60693 CY5CL2 155521553 Ki = 1320 nM T60693 CNO48K 155521726 Ki = 6.4 nM T60693 C70TWB 155522280 Ki = 390 nM T60693 C7QCK2 155522403 EC50 > 10 nM T60693 C10BVP 155522440 Ki = 98 nM T60693 CJP98M 155522548 Ki = 58 nM T60693 CWA8B7 155523094 Ki = 1200 nM T60693 C35CGK 155523518 Ki = 0.78 nM T60693 CQF7N0 155524713 Ki = 1180 nM T60693 C24PLM 155525923 Ki > 1000 nM T60693 C8LIJ9 155526411 Ki = 575 nM T60693 CDFR34 155526934 EC50 = 1.4 nM T60693 C3YE2A 155527040 Ki = 100 nM T60693 CL1N9H 155527202 Ki = 8 nM T60693 C1SZ3R 155527414 IC50 = 0.77 nM T60693 C5B7LS 155527564 Ki = 8.6 nM T60693 CJU69X 155527807 Ki = 410 nM T60693 CO32GB 155528738 EC50 = 174.8 nM T60693 C15MKR 155529017 EC50 = 3.4 nM T60693 CV42PH 155529675 Ki = 1.4 nM T60693 CV1K9L 155529956 Ki = 412 nM T60693 C4G9BP 155530173 EC50 = 2.8 nM T60693 CR1W9V 155530441 Ki = 610 nM T60693 CRYQ39 155530478 EC50 = 0.19 nM T60693 CXH95L 155531153 Ki = 2750 nM T60693 CRZ54B 155532072 Ki < 10000 nM T60693 C6W5JY 155532087 Ki = 4650 nM T60693 C0JF8G 155532588 Ki = 2.2 nM T60693 C68ZHY 155532812 EC50 = 2 nM T60693 C9T0KV 155533432 Ki = 240 nM T60693 CEG3N8 155533730 Ki > 100000 nM T60693 C6GRU2 155533802 Ki = 50.27 nM T60693 CX7TP4 155533942 Ki = 13 nM T60693 CX8DA6 155535193 Ki = 7 nM T60693 CB79ZW 155536080 Ki = 316.23 nM T60693 CR94QG 155536261 Ki = 1550 nM T60693 C08DUJ 155536454 Ki = 16 nM T60693 C2YV1C 155536562 EC50 = 25.9 nM T60693 CE6Q7N 155536593 Ki = 686 nM T60693 C49BUS 155536892 Ki = 20.8 nM T60693 CCO1X2 155537458 Ki = 307 nM T60693 CR97JX 155537513 Ki = 4478 nM T60693 CHLN93 155538528 Ki = 84 nM T60693 CE8UF7 155539181 Ki > 100000 nM T60693 CPDK87 155539216 Ki = 3.2 nM T60693 C5NE1H 155539282 Ki = 37.3 nM T60693 C9S2IA 155539605 Ki = 1707 nM T60693 CX86BV 155539726 Ki = 101 nM T60693 C5E0AD 155540132 Ki = 160 nM T60693 C4G0IA 155540770 Ki = 120.9 nM T60693 C95WGM 155542412 Ki = 8 nM T60693 C67WLH 155542684 Ki > 10000 nM T60693 CI87DG 155543078 Ki = 21.4 nM T60693 CND61A 155543456 Ki = 160 nM T60693 CA27KR 155543816 IC50 = 0.76 nM T60693 C4NI7J 155545136 Ki = 40 nM T60693 CK36RG 155545176 Ki = 9150 nM T60693 CKZ28O 155545411 Ki = 1.1 nM T60693 CFY28C 155545981 Ki = 80 nM T60693 C9QE7K 155546186 Ki = 58.6 nM T60693 CGKR14 155546429 EC50 > 10000 nM T60693 CWE7B0 155549043 Ki = 201 nM T60693 CKAN65 155549973 IC50 = 1.7 nM T60693 CDFU45 155549997 EC50 = 46.7 nM T60693 CJC64E 155551607 Ki = 7.8 nM T60693 C4S7MG 155551744 IC50 = 0.59 nM T60693 C5AQR9 155551873 Ki = 100 nM T60693 C2G7SR 155551876 Ki = 360 nM T60693 CX8JA1 155552185 Ki = 4300 nM T60693 C0WH2Y 155552342 Ki > 100000 nM T60693 C9B5YV 155553316 Ki = 4.3 nM T60693 C81USE 155554575 Ki > 1870 nM T60693 CE2PJ9 155555050 EC50 = 9.7 nM T60693 CM1QS4 155555052 Ki = 53 nM T60693 C91GQI 155555315 Ki = 309.9 nM T60693 C2D5JQ 155555693 Ki = 40 nM T60693 CLB74M 155556900 EC50 = 10 nM T60693 C1ZU4V 155557854 Ki = 1551 nM T60693 CK54XI 155558339 EC50 = 6 nM T60693 CA68FP 155558780 Ki = 89.04 nM T60693 C61BFO 155559678 Ki = 430 nM T60693 CWQ51M 155560805 Ki = 46 nM T60693 C20UAD 155561395 Ki > 100000 nM T60693 C7NO0B 155561575 Ki = 19.5 nM T60693 CZ5Q3J 155562055 EC50 = 1.6 nM T60693 CJT89K 155563204 IC50 = 1.5 nM T60693 CO53GP 155563400 Ki = 1090 nM T60693 CAN0G3 155563660 Ki > 1000 nM T60693 CIS95O 155565113 Ki = 1.8 nM T60693 CEZ16B 155565184 Ki > 100000 nM T60693 CFNC10 155565326 Ki = 2630 nM T60693 CY0N4M 155565847 Ki = 20.3 nM T60693 CUQ25H 155566579 Ki = 293.3 nM T60693 CL76VI 155566581 Ki = 12.4 nM T60693 C23QFO 155567468 Ki = 27 nM T60693 CTNU54 155569410 Ki = 23.2 nM T60693 C57WEG 155569440 Ki = 142 nM T60693 CQ0GL3 155569552 Ki = 674 nM T60693 C3N9VU 10251906 Ki = 288 nM T60693 CP9TR0 10324985 Ki > 10000 nM T60693 CVDX02 13935836 IC50 = 5.5 nM T60693 C9FSE0 14015071 IC50 = 9.1 nM T60693 C13REG 44471685 Ki = 1477 nM T60693 CFR6A5 46905974 Ki = 26 nM T60693 C3C7AZ 49796843 Ki = 0.21 nM T60693 D00FXL 44439907 Ki > 10000 nM T60693 D00JPB 44434951 Ki = 9.6 nM T60693 D00NRB 6602241 Ki = 0.003 nM T60693 D00SDP 44627900 Ki = 0.047 nM T60693 D00TNR 5311081 Ki > 500 nM T60693 D00XZH 44430025 Ki = 7390 nM T60693 D00YCW 44426807 Ki = 245 nM T60693 D01BPI 44456305 EC50 = 26 nM T60693 D01EPU 9804450 Ki = 0.073 nM T60693 D01FPD 44456375 Ki = 1.9 nM T60693 D01HOP 44439875 Ki > 10000 nM T60693 D01MUV 10314141 Ki = 1073 nM T60693 D01RFG 10086063 Ki = 0.06 nM T60693 D01SDX 44439910 Ki > 10000 nM T60693 D01WMU 9820782 Ki = 1712 nM T60693 D02IMZ 44427184 Ki = 0.3 nM T60693 D02NSY 10296561 IC50 = 2500 nM T60693 D02PIG 11250396 Ki = 1030 nM T60693 D02RYZ 16083055 Ki = 0.28 nM T60693 D03KAQ 44626544 Ki = 380 nM T60693 D03PIF 44456106 EC50 = 2.8 nM T60693 D03PTV 10022129 Ki = 488 nM T60693 D03RBD 49765077 IC50 = 20 nM T60693 D03SAV 3082718 Ki = 0.04 nM T60693 D03UFD 5491897 Ki = 396 nM T60693 D03UHT 44429061 Ki = 1.9 nM T60693 D03UJW 22970051 Ki = 4563 nM T60693 D04FBZ 5284595 Ki = 0.38 nM T60693 D04JCJ 44434931 Ki > 5000 nM T60693 D04JCK 644209 Ki = 0.5 nM T60693 D04JFL 16099582 Ki = 0.56 nM T60693 D04PPP 44406697 Ki = 0.076 nM T60693 D04QUB 25242485 Ki = 17 nM T60693 D04TZR 3683 Ki = 2.69 nM T60693 D04UIK 44427178 Ki = 0.046 nM T60693 D04VJE 44434061 Ki > 5000 nM T60693 D04ZQX 44426812 Ki = 335 nM T60693 D05BCY 44425463 EC50 > 2000 nM T60693 D05BZQ 44415858 Ki = 7.9 nM T60693 D05COL 11440685 EC50 = 0.6 nM T60693 D05EWZ 44444966 Ki > 3000 nM T60693 D05EZE 10077295 Ki = 520 nM T60693 D05FEQ 5359966 Ki = 0.034 nM T60693 D05JSY 10462426 Ki = 0.078 nM T60693 D05QJS 5480230 Ki = 0.027 nM T60693 D05RII 44413409 Ki = 330 nM T60693 D05XCV 44583427 Ki > 1000 nM T60693 D05ZIH 45110000 Ki = 7.42 nM T60693 D05ZUX 44207909 Ki >= 1000 nM T60693 D06EES 461776 EC50 = 80 nM T60693 D06EMC 11392888 IC50 = 5800 nM T60693 D06IXE 11411315 Ki = 18 nM T60693 D06KFX 44583372 Ki = 29 nM T60693 D06MQG 44430018 Ki = 3668 nM T60693 D06NST 19143 Ki = 0.07 nM T60693 D06OKE 44427174 Ki = 3.3 nM T60693 D06PHT 10269001 Ki = 364 nM T60693 D06PVO 44426806 Ki = 1427 nM T60693 D06QGJ 52946209 Ki = 75 nM T60693 D06SZI 44429060 Ki = 47 nM T60693 D06TQU 9955378 IC50 = 0.1 nM T60693 D06UTW 44456421 Ki = 5.3 nM T60693 D07BPA 11645313 Ki > 10000 nM T60693 D07CIU 9924923 Ki = 4054 nM T60693 D07DFD 44427176 Ki = 3.4 nM T60693 D07FCB 9925737 Ki = 4149 nM T60693 D07HFU 44429064 Ki = 2.3 nM T60693 D07JIQ 44439882 Ki > 10000 nM T60693 D07KTF 24873526 EC50 = 0.14 nM T60693 D07NMH 10093682 Ki = 2612 nM T60693 D07PPK 44406272 Ki = 126 nM T60693 D07QUY 44583388 Ki = 14 nM T60693 D08DVV 44430026 Ki = 9221 nM T60693 D08IWF 44427180 Ki = 0.81 nM T60693 D08IXN 5497186 Ki = 2.9 nM T60693 D08LIT 11641503 Ki > 1000000 nM T60693 D08QBS 44178080 IC50 = 9800 nM T60693 D08QBU 44430029 Ki = 1801 nM T60693 D08RPH 11255361 Ki = 1.8 nM T60693 D08TFY 10043439 Ki = 387 nM T60693 D08UOX 5281148 Ki = 2515 nM T60693 D08UZJ 12368881 Ki = 78 nM T60693 D09BWX 44583373 Ki = 3.8 nM T60693 D09BYD 20481138 Ki = 818 nM T60693 D09DUE 44429063 Ki = 8.9 nM T60693 D09FJY 9863568 Ki = 802 nM T60693 D09FLC 44627904 Ki = 5.2 nM T60693 D09GQP 15384271 IC50 = 37503 nM T60693 D09LRO 44430008 Ki = 1994 nM T60693 D09RPR 16737207 Ki > 10000 nM T60693 D09RUY 44627790 Ki = 0.34 nM T60693 D09SBU 44583393 IC50 = 5 nM T60693 D09UKS 11303119 Ki = 0.79 nM T60693 D09VRT 44426814 Ki = 288 nM T60693 D09WSG 44456309 Ki = 147 nM T60693 D0A3KA 44456346 Ki = 31 nM T60693 D0A3YH 24853671 Ki > 1000000 nM T60693 D0A9AJ 44439901 Ki > 10000 nM T60693 D0AC0A 10047612 Ki > 400 nM T60693 D0B8MY 9897164 Ki = 0.049 nM T60693 D0C2UQ 44427183 Ki = 0.051 nM T60693 D0C7MP 44429062 Ki = 0.61 nM T60693 D0C9II 45266000 EC50 = 5.7 nM T60693 D0D0UP 10315818 Ki = 3412 nM T60693 D0D5QV 9838803 Ki = 450 nM T60693 D0D5VD 44583375 Ki = 140 nM T60693 D0D6KZ 46906981 Ki = 0.152 nM T60693 D0D8AN 13374610 Ki = 0.24 nM T60693 D0D9BB 10427620 Ki = 13180 nM T60693 D0E0OF 44456378 Ki = 35 nM T60693 D0E0TD 44434950 Ki = 1.22 nM T60693 D0E6GH 44565511 Ki = 0.41 nM T60693 D0E6IT 44439879 Ki > 10000 nM T60693 D0E9HW 44456420 Ki = 2.2 nM T60693 D0ET0T 44425462 EC50 = 123 nM T60693 D0F1EB 44417373 IC50 = 9.81 nM T60693 D0F4AN 44427182 Ki = 4.3 nM T60693 D0F8AX 44430024 Ki = 26405 nM T60693 D0F8CV 5462471 Ki = 270 nM T60693 D0FF6S 16038374 IC50 > 10000 nM T60693 D0G4FA 10384734 Ki = 10298 nM T60693 D0G4NM 104787 Ki > 10000 nM T60693 D0G7DF 44426827 Ki = 1095 nM T60693 D0G7FB 9798655 Ki = 0.049 nM T60693 D0H0KP 44434946 Ki = 45.83 nM T60693 D0H2CI 44456192 EC50 = 0.4 nM T60693 D0H3VZ 44456307 Ki = 13 nM T60693 D0HB6O 44439880 Ki = 1300 nM T60693 D0HN2M 44430609 Ki = 4.365 nM T60693 D0HQ0E 55652 EC50 = 18 nM T60693 D0I1NG 44434058 Ki = 1.15 nM T60693 D0I1ZN 44583428 Ki > 1000 nM T60693 D0I2CE 44583376 Ki = 78 nM T60693 D0I9SX 14707 IC50 = 121 nM T60693 D0IL9H 44430013 Ki = 19695 nM T60693 D0IY2V 44429065 Ki = 20 nM T60693 D0J1PJ 135349 Ki = 0.73 nM T60693 D0J3NK 44427177 Ki = 0.14 nM T60693 D0J5JO 44430009 Ki = 1151 nM T60693 D0J7VL 44439873 Ki > 10000 nM T60693 D0JH5D 44430007 Ki = 1738 nM T60693 D0K1BV 44628003 Ki = 340 nM T60693 D0K3UL 9796720 Ki = 300 nM T60693 D0K4XQ 44427175 Ki = 36 nM T60693 D0L5DN 11392313 Ki = 0.18 nM T60693 D0L5MW 181743 Ki > 10000 nM T60693 D0L6QN 10070040 Ki = 5.5 nM T60693 D0L8LX 123704 Ki = 210 nM T60693 D0L8YY 10066285 Ki = 1.1 nM T60693 D0L9YP 44254503 Ki = 560 nM T60693 D0M9GO 115208 Ki = 0.17 nM T60693 D0N2DN 25129089 Ki = 3400 nM T60693 D0O1JD 44434057 Ki = 18.41 nM T60693 D0O6SB 443408 Ki = 0.02 nM T60693 D0O7JV 44426810 Ki = 220 nM T60693 D0O7RK 44456347 Ki = 141 nM T60693 D0OH7D 5310988 Ki = 28.3 nM T60693 D0P2LE 44596230 IC50 = 1.03 nM T60693 D0P2TT 73354725 Ki > 10000 nM T60693 D0P3FP 44426808 Ki = 36 nM T60693 D0P5IH 44583387 Ki = 66 nM T60693 D0P5QI 44626540 Ki = 40 nM T60693 D0P6FF 44627901 Ki = 2.8 nM T60693 D0P8TI 11466688 Ki = 390 nM T60693 D0PN3P 44439877 Ki > 10000 nM T60693 D0Q3CD 44456105 Ki = 72 nM T60693 D0Q5AJ 44365804 Ki = 120 nM T60693 D0Q6CF 44583374 Ki = 220 nM T60693 D0Q9TQ 10043898 Ki = 343 nM T60693 D0QH4A 10089987 Ki = 759 nM T60693 D0R2VL 44434060 Ki > 5000 nM T60693 D0R4QF 11431898 Ki = 90 nM T60693 D0R5TA 5311080 Ki = 2048 nM T60693 D0R6VF 6540640 IC50 = 0.1 nM T60693 D0R7OE 44456377 Ki = 1.6 nM T60693 D0R9AP 44439872 Ki > 10000 nM T60693 D0S1MA 14376449 Ki = 2600 nM T60693 D0S2OA 10388166 Ki = 13390 nM T60693 D0S3TZ 5748293 EC50 = 117 nM T60693 D0S5FN 44439876 Ki = 2400 nM T60693 D0SC3W 44406704 Ki = 10 nM T60693 D0SE9S 9887077 Ki = 131 nM T60693 D0T2RY 9948320 Ki >= 1000 nM T60693 D0T4ZY 44426817 Ki = 1028 nM T60693 D0T6OQ 10021946 Ki = 0.36 nM T60693 D0T9KE 44430016 Ki = 4160 nM T60693 D0U5OP 11580459 Ki > 10000 nM T60693 D0U7JS 44439866 Ki = 460 nM T60693 D0U7PT 25075996 Ki = 0.0008 nM T60693 D0UG5M 9956146 Ki = 0.01 nM T60693 D0V3OY 105104 Ki = 0.3 nM T60693 D0VO7C 10677974 Ki = 0.059 nM T60693 D0W0CO 44627903 Ki = 1.5 nM T60693 D0W1YD 44439896 Ki > 10000 nM T60693 D0W2DN 44427179 Ki = 0.14 nM T60693 D0W3VT 10091033 Ki = 1702 nM T60693 D0W7DM 17747979 EC50 = 287 nM T60693 D0WT7H 5311018 Ki = 0.94 nM T60693 D0X4SX 10317947 Ki = 1484 nM T60693 D0X5TB 44439905 Ki > 10000 nM T60693 D0XX1Y 44426828 Ki = 2687 nM T60693 D0Y5LJ 10336926 Ki = 9644 nM T60693 D0Y5ZP 44626534 Ki = 280 nM T60693 D0Y7CI 123924 IC50 = 2480 nM T60693 D0Y7KE 44430012 Ki = 11355 nM T60693 D0Y8NO 22977851 Ki = 14.5 nM T60693 D0YU5H 44434949 Ki = 1.78 nM T60693 D0Z8JX 44583386 Ki = 20 nM T60693 D0ZE2W 44430028 Ki = 1438 nM T60693 D0ZG9I 21589297 Ki = 140 nM T78943 D01JUF 5775 Ki = 11.4 nM T78943 D01MDT 5487 Ki = 28.3 nM T78943 D03SKR 2803 Ki = 8.9 nM T78943 D06OFS 68712 Ki = 59.16 nM T78943 D07MOX 439260 Ki > 100000 nM T78943 D09EBS 4636 Ki = 6.194 nM T78943 D0E9PK 4810 IC50 = 3.548 nM T78943 D0K7WK 4595 Ki > 10000 nM T78943 D0L4HY 5702063 Ki = 34.67 nM T78943 D0O6IZ 4436 Ki = 121.6 nM T78943 D0Z2MB 6918107 Ki > 10000 nM T78943 D00OWF 5280953 Ki = 22 nM T78943 C4JQ7T 2068 Ki = 42 nM T78943 COSX53 3519 Ki = 19.01 nM T78943 C32BCH 4656 Ki = 4.797 nM T78943 CL3Q6V 13639 Ki = 39.81 nM T78943 CL34DN 26137 Ki = 1.585 nM T78943 CU86VK 54459 Ki = 7.943 nM T78943 CGW3X5 58533 Ki = 199.53 nM T78943 C3S9TA 58544 Ki = 1.995 nM T78943 C3BQ9D 69591 Ki = 1258.93 nM T78943 CY7ZC9 70319 Ki = 3981.07 nM T78943 CEZ9Q2 71899 Ki = 1.995 nM T78943 C4X7HB 72016 Ki = 52.36 nM T78943 CX17DE 131284 Ki = 231.74 nM T78943 CGT8R0 160510 Ki = 46 nM T78943 CD3ET5 231469 Ki = 7.943 nM T78943 CE5HT0 238079 Ki = 1258.93 nM T78943 COK74Z 345764 Ki = 630.96 nM T78943 C3KM4Y 408156 Ki = 630.96 nM T78943 C4WYR1 594045 Ki = 251.19 nM T78943 C0D5JK 2737433 Ki = 158.49 nM T78943 CUA2H0 3084422 Ki = 31.62 nM T78943 CW04IO 3086495 Ki = 5.012 nM T78943 C1WJ9H 3158580 Ki = 5200 nM T78943 CPCL54 3746427 Ki = 5.012 nM T78943 C98HXL 3771231 Ki = 15.85 nM T78943 C5J1DA 4393018 Ki = 199.53 nM T78943 C6VR5J 6603748 IC50 = 8100 nM T78943 CA51BY 9794143 Ki = 1584.89 nM T78943 C13MBI 9794144 Ki < 10000 nM T78943 C89HIW 9837412 Ki = 10 nM T78943 CB9X7K 9837537 Ki = 1.99 nM T78943 C29SRO 9996353 Ki = 79.43 nM T78943 CUIL41 10012705 Ki = 5.012 nM T78943 C6M4BI 10057802 Ki = 10 nM T78943 CL53TD 10176639 Ki = 537.03 nM T78943 CDOU49 10219780 Ki = 645.65 nM T78943 C0HS9G 10242469 Ki = 7.943 nM T78943 C6Q1DA 10262328 Ki = 10 nM T78943 CL4R3I 10313366 Ki = 512.86 nM T78943 CBYF76 10354045 Ki = 4.7 nM T78943 C5BME0 10374995 Ki = 6.31 nM T78943 C8HWU6 10375456 Ki = 3.162 nM T78943 CUJ32V 10419932 Ki = 11.75 nM T78943 C5DY8H 10442436 Ki = 22.91 nM T78943 CXFE98 10588013 Ki < 10000 nM T78943 C6TFB4 10634173 Ki = 63.1 nM T78943 CF4Y1O 10657832 Ki = 169.82 nM T78943 C0L4QP 10797646 Ki = 331.13 nM T78943 CID3R4 10868559 Ki = 158.49 nM T78943 CZIQ01 10922759 Ki = 10 nM T78943 C8A3LU 10933317 Ki = 470 nM T78943 CT3ZI9 10967219 Ki = 5590 nM T78943 C05XCR 10977777 Ki = 100 nM T78943 CV70ZA 10978438 Ki = 93 nM T78943 CA8Q9Z 10987033 Ki = 1.072 nM T78943 C3VR2W 10997791 Ki = 7244.36 nM T78943 CMU71R 11021868 Ki = 621 nM T78943 CE9T7A 11022127 Ki = 7 nM T78943 C15HYE 11031586 Ki = 3.5 nM T78943 C0A9OC 11031718 Ki = 22.7 nM T78943 CUTM06 11042529 Ki = 31.62 nM T78943 C7Q3ZX 11043404 Ki = 1000 nM T78943 CDIR37 11044324 Ki > 1000 nM T78943 CVB75J 11053968 Ki = 63.1 nM T78943 CJ58RV 11055234 Ki = 560 nM T78943 CJ1QY8 11063180 Ki = 588.84 nM T78943 C0BT2U 11064673 Ki = 43 nM T78943 C5XGY9 11074976 Ki = 10000 nM T78943 CW85AV 11075930 Ki = 140 nM T78943 CT7Q1B 11119320 Ki = 17 nM T78943 CRT6N5 11137887 Ki = 6309.57 nM T78943 CSXV82 11138988 Ki = 47 nM T78943 CGIZ95 11159387 Ki = 6309.57 nM T78943 CL4K0S 11241345 Ki = 50.12 nM T78943 CH2FX9 11747682 Ki = 690 nM T78943 C7LH6B 11770304 Ki = 10000 nM T78943 CAN5Y6 11781522 Ki = 5300 nM T78943 CUB8Q0 12191520 Ki = 100 nM T78943 C78YLK 12248147 Ki = 10000 nM T78943 COYN25 12333190 Ki = 398.11 nM T78943 CPW7N4 12366083 Ki = 10000 nM T78943 C7PEN5 12366096 Ki = 10000 nM T78943 CR1NT6 12632113 Ki = 6025.6 nM T78943 C9GQ4Z 12632114 Ki = 3162.28 nM T78943 CD40XG 12761754 Ki = 3162.28 nM T78943 CKG7B6 12843664 Ki = 7943.28 nM T78943 CNHG28 12863226 Ki = 79.43 nM T78943 CEJ70T 13393069 Ki = 10000 nM T78943 CAK0Y6 13425078 Ki = 50.12 nM T78943 CBTJ50 13425090 Ki = 1584.89 nM T78943 CY97SK 13425094 Ki = 50.12 nM T78943 CMC26O 13869340 Ki = 3.981 nM T78943 C5PD3O 13869343 Ki = 15.85 nM T78943 CQ76WL 14456173 Ki = 10 nM T78943 C7VAQ3 14964720 Ki = 39.81 nM T78943 CCAI21 15407019 Ki = 630.96 nM T78943 CY0NJ5 17774023 Ki = 79.43 nM T78943 C24HWZ 17774025 Ki = 5.012 nM T78943 C8FHS0 17774026 Ki = 39.81 nM T78943 CTD13R 18788392 Ki = 7943.28 nM T78943 CXGA32 19763483 Ki = 158.49 nM T78943 CT84EK 21608213 Ki = 50.12 nM T78943 C2DN1W 21819953 Ki = 25.12 nM T78943 CKIP49 24971933 Ki = 79.43 nM T78943 C21UPD 25883577 Ki = 2.512 nM T78943 C8N7OG 25883581 Ki = 0.7943 nM T78943 CE1Z6D 25883599 Ki = 3.981 nM T78943 C2UX5O 44268929 Ki = 2.512 nM T78943 CZQ54H 44268938 Ki = 1258.93 nM T78943 CO65VL 44269006 Ki = 1.259 nM T78943 C0TP2Z 44269013 Ki = 6.31 nM T78943 CHU5N0 44269016 Ki = 158.49 nM T78943 C5PX3V 44269036 Ki = 63.1 nM T78943 CY01QF 44269044 Ki = 100 nM T78943 C40ZSP 44269051 Ki = 25.12 nM T78943 CUM8P4 44269069 Ki = 10 nM T78943 CR9PJ5 44269074 Ki = 79.43 nM T78943 C6Q8RX 44269086 Ki = 50.12 nM T78943 COB7V3 44269088 Ki = 199.53 nM T78943 CW6A9E 44269089 Ki = 5011.87 nM T78943 C2RWL9 44269090 Ki = 158.49 nM T78943 C7PG8R 44269098 Ki = 398.11 nM T78943 CGQK91 44269099 Ki = 10000 nM T78943 C9T7MG 44269100 Ki = 2.512 nM T78943 CF70OX 44269103 Ki = 79.43 nM T78943 C37XCE 44269105 Ki = 10 nM T78943 CG2D6U 44269106 Ki = 3.981 nM T78943 CPIW69 44269107 Ki = 31.62 nM T78943 CLE3A7 44269115 Ki = 630.96 nM T78943 CZ63DE 44269122 Ki = 309.03 nM T78943 C3I8AT 44269123 Ki = 1995.26 nM T78943 C89FEL 44269124 Ki = 316.23 nM T78943 CFH0C6 44269128 Ki = 3.162 nM T78943 CQZ15X 44269134 Ki = 5011.87 nM T78943 CBS13Z 44269138 Ki = 3162.28 nM T78943 CDS8G5 44269140 Ki = 2511.89 nM T78943 C5SOY3 44269160 Ki = 1000 nM T78943 CN9TV2 44269161 Ki = 39.81 nM T78943 CM57PN 44269162 Ki = 10000 nM T78943 C7V4AB 44302352 Ki > 1000 nM T78943 CS3B6M 44309180 Ki = 17.38 nM T78943 C67ZNM 44352207 Ki = 125.89 nM T78943 CZTA92 44363923 Ki = 37 nM T78943 CIP16C 44403937 Ki = 2022 nM T78943 C13GWS 53821187 Ki = 724.44 nM T78943 CBRI02 78114597 IC50 = 7244.36 nM T78943 CMF3A7 78114671 IC50 = 3388.44 nM T78943 C8JFM6 78114674 IC50 = 8.128 nM T78943 CR6Z8F 78114676 IC50 > 1000000 nM T78943 CTS2P9 78114881 IC50 = 7413.1 nM T78943 C8A6EV 136135852 Ki = 251.19 nM T78943 CAS3E0 155510985 IC50 = 10.47 nM T78943 C75CEX 155513073 IC50 = 1348.96 nM T78943 CVU8Q3 155513359 IC50 = 5495.41 nM T78943 CTV3M6 155521287 Ki = 912000 nM T78943 CK8U7X 155526524 IC50 = 645.65 nM T78943 CD5Y1E 155533747 IC50 = 7585.78 nM T78943 C08RIO 155540329 IC50 = 181.97 nM T78943 CR3T5H 155546767 IC50 = 602559.59 nM T78943 C7V2KX 155547631 IC50 = 28.84 nM T78943 C2EO4B 155567867 IC50 = 64.57 nM T78943 D03LPH 107838 Ki = 180 nM T78943 D04ZPU 11769428 Ki = 0.631 nM T78943 D05GDP 599482 Ki = 12 nM T78943 D05ZUX 44207909 Ki >= 1000 nM T78943 D06BAC 10467319 Ki = 3740 nM T78943 D06QKW 2765 Ki = 3.981 nM T78943 D09BIV 6455104 Ki = 1.995 nM T78943 D09ZDQ 840808 Ki = 2511.89 nM T78943 D0A4AB 2457 Ki = 1.585 nM T78943 D0K8SK 237746 Ki = 5.012 nM T78943 D0LI3J 3080926 Ki = 1.585 nM T78943 D0N9FH 10442227 Ki = 1 nM T78943 D0P4KF 44269078 Ki = 501.19 nM T78943 D0T2RY 9948320 Ki >= 1000 nM T78943 D0Z7NC 33273 Ki = 2.512 nM T68782 D05ZTH 5311181 EC50 = 147 nM T68782 D0N2SR 9913767 EC50 = 100 nM T68782 D0WL5V 9867642 IC50 = 0.09 nM T68782 D00HTY 5280363 IC50 = 4500 nM T68782 D00MZK 9911469 Ki = 2300 nM T68782 D0GC5H 123879 Ki > 10000 nM T68782 D0I3TU 45268455 Ki = 373 nM T68782 D0K1EG 11508736 IC50 > 10000 nM T68782 D0M4TJ 44219292 EC50 = 850 nM T68782 D0RL4X 45270144 IC50 = 25600 nM T68782 D0SP5V 49843471 IC50 = 1290 nM T68782 D0X7EG 11462174 IC50 = 7300 nM T68782 D0YB2Y 42641863 IC50 = 35 nM T68782 D0K0VH 9867949 IC50 = 0.4 nM T68782 CYFR68 5036 Ki = 6140 nM T68782 C3W5UX 7204 Ki > 10000 nM T68782 CFG9T5 1101166 IC50 > 10000 nM T68782 CLM8P6 2114670 Ki > 25000 nM T68782 CO7N1Z 5311239 IC50 > 10000 nM T68782 CM4AB0 6461002 Ki > 10000 nM T68782 CB5DJ4 7097680 IC50 > 10000 nM T68782 CURH60 9801972 Ki = 1.8 nM T68782 CQA35F 9802748 Ki = 6100 nM T68782 CGC14Q 9803349 IC50 = 0.9 nM T68782 C6TA3N 9809136 Ki = 2400 nM T68782 CV24TI 9817292 Ki = 4100 nM T68782 CHUM01 9825028 Ki = 4 nM T68782 CXI27J 9872340 IC50 = 55 nM T68782 CKMW12 9874010 Ki = 2870 nM T68782 CF0HC5 9888589 IC50 > 10000 nM T68782 CFC8G4 9894720 Ki > 3000 nM T68782 CA5N0K 9895436 Ki = 4000 nM T68782 CKNG97 9931891 EC50 = 154 nM T68782 CZ5Q3U 9933925 Ki = 9.5 nM T68782 CICE70 9938626 Ki = 2800 nM T68782 CWDT69 9939791 Ki = 2000 nM T68782 C6SGH7 9954562 Ki > 500 nM T68782 C4UK2Q 9955802 Ki > 3000 nM T68782 CKIE37 9985715 IC50 = 16000 nM T68782 CMPT81 10025456 IC50 = 22 nM T68782 CHN98V 10028338 Ki = 1.3 nM T68782 CQ3GW6 10047541 IC50 > 10000 nM T68782 CM89DR 10073359 Ki = 3.7 nM T68782 CV48SW 10074101 Ki = 1.8 nM T68782 C6NT2P 10098978 IC50 = 13 nM T68782 CEX2R1 10116114 IC50 = 1.2 nM T68782 CEM21G 10181606 Ki = 830 nM T68782 CB59SL 10183680 IC50 = 10 nM T68782 CTGL49 10206535 IC50 = 0.81 nM T68782 CB7XJ2 10216985 Ki = 0.89 nM T68782 C0ED9Y 10251023 IC50 > 10000 nM T68782 C8YHK7 10254794 Ki = 1.3 nM T68782 CL7YG3 10287121 Ki > 13000 nM T68782 CM7E1S 10342667 Ki = 6 nM T68782 CWT1K9 10344683 Ki = 1.4 nM T68782 CM1VU7 10345671 Ki = 3.3 nM T68782 CB19MW 10402929 Ki = 2400 nM T68782 CRFZ84 10432190 Ki = 12.4 nM T68782 CGT5X1 10433093 Ki = 0.39 nM T68782 CHW12E 10458032 Ki = 3.7 nM T68782 CC83QY 10480515 Ki = 1.9 nM T68782 CZ1XW6 10483360 IC50 = 12 nM T68782 CYTV60 10502508 IC50 = 26 nM T68782 C39BYU 10502610 IC50 = 420 nM T68782 CZ2H8E 10529261 IC50 = 780 nM T68782 C4F9MA 10529683 IC50 = 1300 nM T68782 CANM20 10547489 IC50 = 38 nM T68782 CTY02L 10552450 IC50 = 380 nM T68782 C58ZOU 10552612 IC50 = 210 nM T68782 C0D7EI 10553794 IC50 = 57 nM T68782 CMO37F 10594576 IC50 = 32 nM T68782 C3GKS1 10595288 IC50 = 360 nM T68782 CJ7IT3 10599289 IC50 = 1.3 nM T68782 CMY4P3 10601359 IC50 = 27 nM T68782 CPV7D6 10623568 IC50 = 450 nM T68782 CD13GN 10648014 IC50 = 570 nM T68782 CI5HA0 10648334 IC50 > 10000 nM T68782 C9YQG5 10670992 IC50 > 10000 nM T68782 C9SUW2 10671942 IC50 = 70 nM T68782 CP1Z8W 10694649 IC50 > 1000 nM T68782 C3WRM7 10696132 IC50 = 320 nM T68782 C7H8NA 10717385 IC50 > 1000 nM T68782 C7GY6X 10739351 IC50 > 10000 nM T68782 CY8IB2 10740699 IC50 > 10000 nM T68782 C12SBH 10741017 IC50 > 10000 nM T68782 CG17HE 10741197 IC50 > 10000 nM T68782 CK8O4Z 10741899 IC50 = 1.8 nM T68782 C64MLE 10767455 IC50 = 47 nM T68782 CD1YX8 10813802 IC50 = 220 nM T68782 C2NVU7 10864153 IC50 = 34 nM T68782 CV80AK 10874325 IC50 = 160 nM T68782 CJMI82 10874343 IC50 = 120 nM T68782 C3IOP0 10874929 IC50 = 33 nM T68782 CT5ZI4 10885356 IC50 = 200 nM T68782 C50EQZ 10885393 IC50 = 90 nM T68782 C4RU1C 10896473 IC50 = 18 nM T68782 CV2Z4D 10917396 IC50 = 280 nM T68782 CA2WX0 10928987 IC50 = 450 nM T68782 CCDR06 10939814 IC50 = 180 nM T68782 CG54WH 10951130 IC50 = 180 nM T68782 CQO6L0 10951507 IC50 = 57 nM T68782 CGD4L9 10961839 IC50 = 100 nM T68782 C4MY1P 10961840 IC50 = 180 nM T68782 C2O1NE 10962613 IC50 = 32 nM T68782 C2GD8P 11004079 IC50 = 390 nM T68782 C54SIX 11005555 IC50 = 120 nM T68782 CUD0T4 11005693 IC50 = 190 nM T68782 CN06LF 11014665 IC50 > 1000 nM T68782 C3G9DR 11026912 IC50 = 580 nM T68782 CTPC12 11037643 IC50 > 1000 nM T68782 C0GYC7 11037976 IC50 > 1000 nM T68782 C26HEW 11038515 IC50 = 36 nM T68782 CIN82G 11059671 IC50 = 200 nM T68782 CGZH23 11059915 IC50 = 530 nM T68782 CY81OU 11070932 IC50 = 64 nM T68782 C9LM7B 11071097 IC50 = 34 nM T68782 CLSJ01 11081109 IC50 > 1000 nM T68782 CP4X5R 11081118 IC50 = 22 nM T68782 CRKE27 11091552 IC50 > 1000 nM T68782 CL9ZS0 11091707 IC50 = 340 nM T68782 CQ09UT 11102462 IC50 = 8600 nM T68782 CA4MQ6 11103335 IC50 = 380 nM T68782 CKST02 11122314 IC50 > 10000 nM T68782 C20WJL 11123691 IC50 > 1000 nM T68782 C6NT1W 11123848 IC50 = 210 nM T68782 CQJL60 11123892 IC50 = 86 nM T68782 C30CRJ 11134066 IC50 = 47 nM T68782 CTL21Y 11134192 IC50 = 670 nM T68782 CFVP96 11134618 IC50 = 1300 nM T68782 C1TSD6 11135113 IC50 = 660 nM T68782 CM8Q9D 11145780 IC50 = 15 nM T68782 CRI92F 11189801 Ki = 2.1 nM T68782 CNU4B3 11245359 Ki > 10000 nM T68782 C4S5MX 11249458 Ki > 10000 nM T68782 CIH90K 11259797 Ki = 0.75 nM T68782 C70ESM 11269563 Ki = 1.1 nM T68782 CW3IZ0 11270709 Ki = 3.6 nM T68782 C9E4SW 11294166 Ki = 1.8 nM T68782 CBJ75S 11294992 Ki = 0.39 nM T68782 C92FAZ 11301859 Ki > 10000 nM T68782 CJ90WI 11386109 Ki = 0.36 nM T68782 CN2TG7 11387144 Ki > 1000 nM T68782 CK7D1E 11407637 Ki > 10000 nM T68782 CXPO04 11408533 Ki = 2.6 nM T68782 C0SLC1 11409320 IC50 = 4.4 nM T68782 CORM68 11485353 Ki > 10000 nM T68782 CE2JA4 11488860 Ki = 0.43 nM T68782 C4QUK1 11494321 Ki = 6890 nM T68782 CW3YO5 11494768 IC50 > 10000 nM T68782 C1IX3W 11495368 IC50 = 6.026 nM T68782 CHPQ36 11495480 IC50 = 7.586 nM T68782 CV72QC 11501025 IC50 = 54.95 nM T68782 CBQX60 11502516 IC50 = 2.884 nM T68782 C3S9HX 11502665 IC50 = 12.88 nM T68782 CQ6IU7 11509269 IC50 = 8200 nM T68782 CDV2U8 11516699 IC50 = 7.079 nM T68782 CB18VF 11517351 IC50 = 100000 nM T68782 C9FQW8 11537884 Ki > 10000 nM T68782 CF2OM8 11539410 IC50 = 780 nM T68782 C4W6IN 11540010 IC50 = 0.01995 nM T68782 C2B8HY 11545850 Ki = 5300 nM T68782 CWB93I 11567324 IC50 = 10.96 nM T68782 CN1O9M 11573030 Ki > 10000 nM T68782 CXQD46 11573799 Ki = 4860 nM T68782 C7XOF0 11582363 IC50 = 7.244 nM T68782 CV0G6S 11584210 IC50 = 0.05012 nM T68782 CM7S6Q 11588648 Ki > 10000 nM T68782 C7Y6XJ 11597294 IC50 = 0.26 nM T68782 CM8H4W 11597347 IC50 = 660.69 nM T68782 C2M8HZ 11610353 IC50 > 10000 nM T68782 CG2JS0 11619108 IC50 = 32.36 nM T68782 CORL03 11625836 Ki = 1872 nM T68782 CN5HP4 11631233 IC50 = 7.762 nM T68782 C9L5VD 11631813 IC50 > 10000 nM T68782 CPY0R4 11639470 IC50 = 41.69 nM T68782 CPR87V 11640888 IC50 = 14.13 nM T68782 CB1EX5 11646256 IC50 = 218.78 nM T68782 C5LI7P 11647012 IC50 > 100000 nM T68782 CMB6F9 11653874 IC50 = 780 nM T68782 C2T7GK 11660493 IC50 = 0.8913 nM T68782 CJ4P0D 11667039 Ki = 6400 nM T68782 C1A4UW 11667189 IC50 = 7.943 nM T68782 C51UDK 11667741 IC50 > 10000 nM T68782 C2C7FO 11668164 IC50 = 64.57 nM T68782 CIV0C5 11669780 IC50 = 0.302 nM T68782 CIUJ01 11670392 IC50 > 10000 nM T68782 C97FRY 11675335 Ki = 8460 nM T68782 C72BNQ 11682521 IC50 > 10000 nM T68782 CW8RY9 11689895 IC50 > 10000 nM T68782 CDJ8H1 11690028 IC50 = 2.291 nM T68782 C9CM2R 11695689 IC50 > 10000 nM T68782 C3BSV4 11696697 Ki > 13000 nM T68782 CH4P6U 11696919 IC50 = 0.3981 nM T68782 CKXG13 11697378 IC50 = 2.57 nM T68782 C4AS6M 11717784 Ki = 7710 nM T68782 C45MZJ 11717787 IC50 = 12.88 nM T68782 C0SQJ4 11717959 IC50 = 0.7943 nM T68782 CZP19Q 11718798 IC50 = 43.65 nM T68782 CLVO97 11733560 IC50 = 260 nM T68782 CAB5I6 11741746 Ki = 0.71 nM T68782 C5QS6Y 11742649 Ki = 16.3 nM T68782 C3OW1Z 11743676 Ki = 0.53 nM T68782 CU21FT 11762410 IC50 = 22 nM T68782 C2HL4F 11811847 IC50 = 130 nM T68782 CKWZ21 11812883 IC50 = 19 nM T68782 CB15GD 11826199 IC50 = 720 nM T68782 C97TPZ 11826761 IC50 = 650 nM T68782 CCB54R 12341157 Ki > 10000 nM T68782 CT34LO 13230981 Ki > 13000 nM T68782 CO19GA 14372497 Ki = 11 nM T68782 C93KFC 14372503 Ki = 80 nM T68782 C69REM 14372504 Ki = 1 nM T68782 CC68GR 14372505 Ki = 2.8 nM T68782 CBD64J 15157534 Ki = 36 nM T68782 CHW6G0 15157538 Ki = 2.6 nM T68782 CB8ZE9 15157541 Ki = 1.7 nM T68782 C29LSJ 15458814 IC50 = 5.6 nM T68782 C06OGJ 15486805 IC50 = 3100 nM T68782 C0L3VU 15486806 IC50 > 10000 nM T68782 CWQ8B9 15551228 Ki > 500 nM T68782 CIS83K 15947857 Ki = 53 nM T68782 C3L0RK 15948325 Ki = 1200 nM T68782 CHBE61 15949677 IC50 > 30000 nM T68782 CM7J9N 16049493 Ki = 1.7 nM T68782 CRZT49 16222207 IC50 = 8500 nM T68782 CI61TE 16678098 IC50 > 31622.78 nM T68782 CNCB74 16681720 Ki = 1.1 nM T68782 CK69TB 18476686 Ki = 1.7 nM T68782 CGF28X 21019821 Ki = 0.38 nM T68782 CX08BC 21198692 Ki = 82 nM T68782 CGU36V 21974328 Ki = 30 nM T68782 CC7SX4 21974362 Ki = 390 nM T68782 C5O4RB 21974374 IC50 = 30 nM T68782 C7YLR9 21974448 IC50 = 250 nM T68782 CGT9U1 21974528 Ki = 20 nM T68782 CPMI48 22083972 Ki = 8.5 nM T68782 CBW0P7 22083975 Ki = 1100 nM T68782 C4SVP2 22083978 Ki = 4.5 nM T68782 CZ5XJ8 22225815 Ki = 1.3 nM T68782 CF81SW 23582412 IC50 > 10000 nM T68782 CP2S4J 23663736 Ki = 2900 nM T68782 C42LYP 24765153 IC50 = 0.22 nM T68782 CF72YI 24765671 Ki = 885 nM T68782 C31JZP 24765672 Ki = 16 nM T68782 C4QX7Y 24765675 Ki = 14 nM T68782 CF4EN6 24765766 Ki = 1205 nM T68782 CL7Z9U 24765768 Ki = 63 nM T68782 CE1K3P 24765769 Ki = 450 nM T68782 CLS5J9 24776302 IC50 > 30000 nM T68782 C4BD1L 24776306 IC50 > 30000 nM T68782 CFQA40 24952577 Ki > 7282 nM T68782 CD98IN 24952580 Ki > 456 nM T68782 C81WVN 24952927 Ki > 5474 nM T68782 CZT83E 24952928 Ki > 501 nM T68782 C8YHX3 24953283 Ki > 224 nM T68782 CZ93FO 24953285 Ki > 628 nM T68782 C17JTY 24953286 Ki > 2226 nM T68782 CFT0W5 24953624 Ki > 4992 nM T68782 C42VMD 24953625 Ki > 3461 nM T68782 C7B2EW 24953628 Ki > 2117 nM T68782 C05VGF 24961406 IC50 > 1000 nM T68782 CXQJ67 25002382 Ki = 561 nM T68782 CN5SH9 25003075 Ki = 1648 nM T68782 CDR8B5 25106870 IC50 = 1100 nM T68782 CQSC30 25106871 IC50 = 27 nM T68782 CEX34J 25817650 Ki = 1115 nM T68782 CO46CI 25908688 Ki > 10000 nM T68782 CG9F0D 25908691 Ki = 4490 nM T68782 CI90SE 35028115 Ki = 9.6 nM T68782 CZG4X7 44128594 IC50 = 14 nM T68782 CNOF71 44138108 IC50 = 0.14 nM T68782 C5G4LN 44159411 IC50 = 36400 nM T68782 CHI65U 44159530 IC50 = 4000 nM T68782 CMNH53 44159772 IC50 = 4000 nM T68782 CUE81M 44188793 IC50 > 50000 nM T68782 C2AV1K 44190762 IC50 = 8450 nM T68782 CZ29JY 44205724 IC50 = 31300 nM T68782 C0A4TB 44232564 EC50 = 1140 nM T68782 C46VMC 44232565 EC50 = 808 nM T68782 CUL10P 44232568 EC50 > 10000 nM T68782 CTK9I3 44233521 EC50 = 860 nM T68782 CQ13MH 44234032 Ki = 1850 nM T68782 C5D2AV 44234532 EC50 = 355 nM T68782 C6B7YM 44234782 EC50 = 1720 nM T68782 CVL8A5 44235044 EC50 = 240 nM T68782 CMG1Y5 44235291 EC50 = 5070 nM T68782 CVBY63 44235519 EC50 = 320 nM T68782 CMJ1G3 44235520 EC50 = 620 nM T68782 CS5CZ3 44235521 EC50 = 2050 nM T68782 C9T5SL 44235522 EC50 > 10000 nM T68782 CM3L2H 44235755 EC50 = 5000 nM T68782 CY76GT 44236221 EC50 = 1030 nM T68782 CR68BA 44250281 Ki > 10000 nM T68782 CN90FE 44269464 Ki > 13000 nM T68782 C1L0ET 44269468 Ki > 13000 nM T68782 C5KRQ4 44269486 Ki > 13000 nM T68782 CL6M2P 44269516 Ki > 13000 nM T68782 CON8R9 44269520 Ki > 13000 nM T68782 C6MBG0 44269521 Ki > 13000 nM T68782 CZ3Q1L 44269523 Ki > 13000 nM T68782 CRL61O 44269532 Ki > 13000 nM T68782 C1Z4LU 44269540 Ki > 13000 nM T68782 CM72FA 44269542 Ki > 13000 nM T68782 CN0JV2 44269543 Ki > 13000 nM T68782 C28UJH 44269544 Ki > 13000 nM T68782 CR1IY6 44269568 Ki > 13000 nM T68782 CI3C9O 44269596 Ki > 13000 nM T68782 CC0EW9 44269597 Ki > 13000 nM T68782 CCG6V3 44344457 IC50 = 460 nM T68782 CLN63A 44377464 Ki = 2500 nM T68782 CK4QD9 44394380 Ki = 10 nM T68782 CUVG09 44394432 Ki = 130 nM T68782 CWL1X4 44400355 Ki > 1000 nM T68782 CJ1O3D 44411552 Ki = 4.1 nM T68782 C2UQV7 44411555 Ki = 1 nM T68782 CNM76B 44411567 Ki = 110 nM T68782 C69PSX 44411605 Ki = 2.8 nM T68782 CE3J1V 44411606 Ki = 9.7 nM T68782 C7MCE5 44411635 Ki = 1900 nM T68782 C8ZUQ5 44411688 Ki = 1.9 nM T68782 C4AD5K 44411791 Ki = 6.3 nM T68782 CZ0X3F 44411797 Ki = 4 nM T68782 CUQ76I 44411798 Ki = 23 nM T68782 CE49GA 44411799 Ki = 4.4 nM T68782 CLH8R3 44411809 Ki = 16 nM T68782 CH7UG4 44411813 Ki = 29 nM T68782 CRP5N3 44411814 Ki = 3.5 nM T68782 CCH0L3 44411851 Ki = 4.1 nM T68782 C5GD6H 44411889 Ki = 28 nM T68782 CO41IV 44411890 Ki = 3.9 nM T68782 COMS38 44411896 Ki = 300 nM T68782 C40QDV 44411984 Ki = 7.5 nM T68782 CIB2W5 44419347 Ki > 500 nM T68782 C91JXT 44419374 Ki > 500 nM T68782 CNF4W2 44419379 Ki > 500 nM T68782 CND06K 44441186 Ki > 10000 nM T68782 C1OKM8 44441196 Ki = 1210 nM T68782 CIV84R 44460415 IC50 = 190 nM T68782 C48SBE 44460432 IC50 > 1000 nM T68782 CWB70V 44460460 IC50 = 320 nM T68782 CLKS48 44460682 IC50 = 73 nM T68782 C41VGA 44460691 IC50 = 170 nM T68782 C7C3DU 44460692 IC50 = 15 nM T68782 CK64GF 44460702 IC50 = 6000 nM T68782 CK9SB3 44460703 IC50 = 500 nM T68782 C7CAV4 44460705 IC50 = 330 nM T68782 C1Q0PH 44460716 IC50 > 1000 nM T68782 C1A5DT 44460730 IC50 = 110 nM T68782 CC4XV0 44460740 IC50 = 3400 nM T68782 C71SGU 44460751 IC50 = 37 nM T68782 C6RA3M 44460813 IC50 = 110 nM T68782 C3X0YS 44460814 IC50 = 25 nM T68782 CM0W9B 44460832 IC50 = 42 nM T68782 CDP24A 44460923 IC50 = 17 nM T68782 C3QDF8 44460938 IC50 = 30 nM T68782 CDR8G2 44460939 IC50 = 18 nM T68782 CVW2T3 44460942 IC50 = 38 nM T68782 C8ZV1H 44460945 IC50 = 93 nM T68782 CU4BO7 44460960 IC50 = 4500 nM T68782 CL5P9E 44460962 IC50 = 180 nM T68782 C5SBH6 44461024 IC50 = 110 nM T68782 C7U9DL 44461046 IC50 = 0.42 nM T68782 C02CUY 44461047 IC50 = 76 nM T68782 C6H8GE 44461053 IC50 = 22 nM T68782 C3W1BR 44461054 IC50 > 10000 nM T68782 CY96TB 44461071 IC50 = 19 nM T68782 CON1M0 44461073 IC50 > 1000 nM T68782 C5K0NL 44461194 IC50 = 35 nM T68782 C32VIB 44461195 IC50 = 74 nM T68782 C95VML 44461209 IC50 = 56 nM T68782 CZY53M 44591457 Ki = 0.88 nM T68782 CJUX12 44591458 Ki = 13.6 nM T68782 C5ZRQ7 44591477 Ki = 1 nM T68782 CFI4O5 44591512 Ki = 1 nM T68782 C87ZCK 44591513 Ki = 0.91 nM T68782 CH2W6M 44591514 Ki = 2.5 nM T68782 CI5SP2 44591515 Ki = 0.8 nM T68782 COH31P 44591516 Ki = 1 nM T68782 CH7LE5 44591535 Ki = 0.74 nM T68782 CZ2UO0 44591536 Ki = 1.14 nM T68782 C4DJH3 44591537 Ki = 0.88 nM T68782 CF5O6R 44591561 Ki = 1.2 nM T68782 CMZ6B3 44591562 Ki = 0.67 nM T68782 C6Z2MX 44591563 Ki = 0.39 nM T68782 CD9KX4 44591762 Ki = 1.6 nM T68782 CJ6S7Q 44591806 Ki = 107.4 nM T68782 CT0L2W 44591807 Ki = 2.3 nM T68782 CRA6S0 45109984 Ki > 12000 nM T68782 C3JE7N 45109987 Ki > 10000 nM T68782 CA28PL 45109988 Ki > 4000 nM T68782 CN6P8B 45109989 Ki > 4000 nM T68782 CY2BK4 45110108 Ki > 4000 nM T68782 CR1KP4 45110109 Ki > 4000 nM T68782 CR6UW4 45112038 Ki > 38000 nM T68782 CULJ91 45268456 IC50 = 31000 nM T68782 CB5O6V 45269307 IC50 = 2200 nM T68782 C03ETI 45270148 IC50 = 9000 nM T68782 CY70SI 45270983 IC50 > 100000 nM T68782 C2XH3A 45270987 IC50 > 100000 nM T68782 C35DUQ 45272700 IC50 = 4400 nM T68782 CKUI32 45272704 IC50 = 37800 nM T68782 C3U7KT 45273637 Ki > 1300 nM T68782 C4XE5C 45486009 IC50 = 9 nM T68782 C0L5AY 45486021 IC50 = 41 nM T68782 C3Y7KG 45486025 IC50 = 43 nM T68782 C2UZP0 45486026 IC50 = 120 nM T68782 CR7YG5 45486030 IC50 = 11 nM T68782 C14LAV 45486038 IC50 = 179 nM T68782 CLO03H 45486043 IC50 = 8300 nM T68782 CE3V7H 45486045 IC50 > 10000 nM T68782 CX0AO7 45486053 IC50 = 132 nM T68782 C1YRG8 45486054 IC50 = 36 nM T68782 CHK46L 45486059 IC50 = 2070 nM T68782 CD6XC5 45486065 IC50 = 36 nM T68782 CK4ZB3 45486073 IC50 > 10000 nM T68782 CF24XK 45486074 IC50 = 31 nM T68782 C7QEA3 45486099 IC50 = 1910 nM T68782 CRCS08 45486100 IC50 = 59 nM T68782 C6RV7G 46701878 IC50 > 1000 nM T68782 C90NLX 46853755 Ki = 1580 nM T68782 C2L3DI 46879343 IC50 > 10000 nM T68782 CI3RS4 46879377 IC50 > 10000 nM T68782 C0A2CI 46890616 Ki = 404 nM T68782 CW52VH 46890658 Ki = 49 nM T68782 CXQ2W0 46890659 Ki = 1389 nM T68782 CQ20RC 46890660 Ki = 209 nM T68782 CTR7Q0 49850345 IC50 > 50118.72 nM T68782 CZ9UD6 50901657 IC50 = 26700 nM T68782 C8VNM2 51003549 Ki > 47000 nM T68782 COZ42H 51031012 IC50 = 5200 nM T68782 C9UO5T 51347010 IC50 > 50000 nM T68782 CVCQ34 51347011 IC50 > 50000 nM T68782 CN80GS 51347012 IC50 > 50000 nM T68782 CJD25G 52920263 IC50 = 19000 nM T68782 C3XYP8 52941281 Ki = 0.36 nM T68782 C6SPT4 52943623 Ki = 0.33 nM T68782 CE04FW 52944928 Ki = 0.33 nM T68782 CA41UT 52944959 Ki = 0.51 nM T68782 CX8L6T 52945002 Ki = 16.5 nM T68782 C9WUH5 52948543 Ki = 0.41 nM T68782 CI8TP9 52948585 Ki = 0.31 nM T68782 CK9DR7 52949846 Ki = 0.38 nM T68782 CTU93P 53316532 Ki > 3400 nM T68782 CRUM06 53316574 IC50 = 0.5012 nM T68782 CAR8G2 53316575 IC50 = 0.5012 nM T68782 C4P2CV 53316653 Ki = 2093 nM T68782 CS4G5H 53316671 Ki = 121 nM T68782 CL96IZ 53316672 Ki = 51 nM T68782 CBT1P4 53316673 Ki > 3901 nM T68782 C7GEO9 53317523 IC50 = 245.47 nM T68782 C8D7UQ 53317569 Ki = 48 nM T68782 C1CFU7 53317642 Ki = 322 nM T68782 CXV3W2 53317718 Ki = 2292 nM T68782 C0ZH3X 53317854 Ki > 3700 nM T68782 C5PC0V 53317886 IC50 = 7.079 nM T68782 CRD12W 53317887 IC50 = 104.71 nM T68782 CEO6D8 53317912 IC50 = 6.31 nM T68782 CP14EK 53317957 Ki = 248 nM T68782 C97LDX 53317958 Ki = 104 nM T68782 C5WO9J 53317977 Ki = 537 nM T68782 CHR16U 53318738 IC50 = 2.291 nM T68782 C6SPD5 53319215 IC50 = 549.54 nM T68782 C1TE9Z 53319216 IC50 = 0.3981 nM T68782 COJ82D 53319320 Ki = 541 nM T68782 C4T9BV 53319321 Ki = 14.6 nM T68782 CE86AP 53319322 Ki = 26 nM T68782 C6UY8I 53320268 IC50 = 3.802 nM T68782 CN79KA 53320526 IC50 = 0.3981 nM T68782 CK5PA0 53320527 IC50 = 0.302 nM T68782 CV8M5K 53320594 Ki = 2391 nM T68782 CZL85A 53320595 Ki = 284 nM T68782 C8EO2U 53320616 Ki = 1282 nM T68782 C5HY9K 53320617 Ki = 1213 nM T68782 CZ40CV 53320618 Ki = 283 nM T68782 C0VWB8 53321438 IC50 = 22.91 nM T68782 CIU6E0 53321678 Ki = 16 nM T68782 CYR51J 53321679 IC50 = 38.02 nM T68782 C7D5BN 53321784 Ki > 12000 nM T68782 C5QOI8 53321785 Ki > 18000 nM T68782 C5MFX6 53321836 IC50 = 1698.24 nM T68782 CQE8T4 53321837 IC50 = 3.631 nM T68782 CF3D7W 53321838 IC50 = 6.026 nM T68782 CY0K2D 53321839 IC50 = 5.012 nM T68782 C89DLV 53321923 Ki = 5.6 nM T68782 C29QNI 53321924 Ki = 47 nM T68782 CJ7C4U 53321925 Ki = 799 nM T68782 CB5S0H 53322785 Ki = 15.5 nM T68782 CLC5O4 53323151 IC50 = 2.692 nM T68782 C8ZM7P 53323152 IC50 = 40.74 nM T68782 C4TU3V 53323153 IC50 = 12.02 nM T68782 CLH52C 53323184 IC50 = 5.129 nM T68782 CPI3O6 53323246 Ki = 216 nM T68782 C2KRB3 53323266 Ki = 711 nM T68782 CMK0A1 53323267 Ki > 4069 nM T68782 C4ZP8Y 53323268 Ki = 130 nM T68782 CTOY32 53324111 Ki = 123 nM T68782 CE23YH 53324462 Ki > 3800 nM T68782 C2OPC0 53324506 IC50 = 0.1 nM T68782 C3YTB9 53324508 IC50 = 8.128 nM T68782 CXVT21 53324509 IC50 = 213.8 nM T68782 C7SLG2 53324534 IC50 = 2.57 nM T68782 CD1GX3 53324544 IC50 = 25.7 nM T68782 CF9SZ3 53324589 Ki = 395 nM T68782 C68JYF 53325826 IC50 = 5.012 nM T68782 CSD80K 53325827 IC50 = 10 nM T68782 CCP07V 53325847 IC50 = 0.5012 nM T68782 C5FWU7 53325848 IC50 = 245.47 nM T68782 CUS37X 53325907 Ki > 3952 nM T68782 CZ1SE0 53325908 Ki = 1079 nM T68782 CH8S3T 53325909 Ki = 892 nM T68782 C9DR3V 53325910 Ki = 1075 nM T68782 CZ7WN5 53325911 Ki = 250 nM T68782 CEMU31 53325912 Ki > 3901 nM T68782 C2R6NQ 53326808 IC50 = 1071.52 nM T68782 CAL29U 53326879 Ki > 3235 nM T68782 CZID32 53495002 IC50 > 10000 nM T68782 C9HK6G 54582728 Ki > 1000 nM T68782 C2RJM1 54583706 Ki > 1000 nM T68782 CGC46Y 54764763 IC50 = 8.1 nM T68782 CR4U7M 56665068 IC50 > 50 nM T68782 CWR1Z7 56665984 Ki > 13000 nM T68782 CD32NT 56834987 IC50 > 10000 nM T68782 CO65JY 56834988 IC50 = 12 nM T68782 C6H2JT 56834989 IC50 = 3 nM T68782 C1U7XJ 56924869 IC50 = 12600 nM T68782 CT4SR8 57335620 IC50 = 10 nM T68782 C4BHP5 57335749 IC50 = 4 nM T68782 CRH1K9 57390757 IC50 = 83 nM T68782 C9BF1I 57390758 IC50 = 5 nM T68782 C2MX5W 57391065 IC50 = 280 nM T68782 CC4UT1 57391066 IC50 = 19 nM T68782 CM41FU 57391518 IC50 > 10000 nM T68782 CJ5OT4 57391799 IC50 = 450 nM T68782 CI56TU 57391800 IC50 = 6 nM T68782 C37ERY 57392564 IC50 = 6 nM T68782 CWZ92U 57392565 IC50 = 630 nM T68782 C53WSX 57392566 IC50 > 10000 nM T68782 CC9V5H 57392567 IC50 > 10000 nM T68782 C3KR1M 57392568 IC50 = 23 nM T68782 C95WXD 57393270 IC50 > 10000 nM T68782 C3MXN1 57393532 IC50 = 8 nM T68782 CXR6Y8 57393533 IC50 = 15 nM T68782 C4FAZ8 57394587 IC50 = 6.5 nM T68782 CQ2J9O 57395244 IC50 = 190 nM T68782 C7IL8F 57395245 IC50 = 310 nM T68782 CO8BR1 57395246 IC50 = 10 nM T68782 C81FYQ 57396042 IC50 = 480 nM T68782 CBR0J8 57396043 IC50 = 230 nM T68782 CQ9OG2 57396044 IC50 = 29 nM T68782 C5GBP8 57396745 IC50 = 910 nM T68782 CDGC05 57396746 IC50 = 7 nM T68782 CW5O7V 57396747 IC50 > 10000 nM T68782 CZ1BY9 57396754 IC50 > 10000 nM T68782 CP5K2O 57397014 IC50 > 10000 nM T68782 C04AJG 57397843 IC50 = 10 nM T68782 C74WUG 57398523 IC50 = 570 nM T68782 C2BLJ3 57398777 IC50 = 21 nM T68782 CD2FV3 57398778 IC50 = 600 nM T68782 CE4VT0 57400453 IC50 = 930 nM T68782 C4DJQ2 57400454 IC50 = 2340 nM T68782 C3K7LZ 57400455 IC50 = 30 nM T68782 C3PGK2 57400456 IC50 = 13 nM T68782 C0BFW6 57400457 IC50 = 20 nM T68782 C5Q7VD 57401263 IC50 = 15 nM T68782 C3DCU4 57401983 IC50 = 6 nM T68782 CJTF24 57402257 IC50 = 9 nM T68782 CYE63U 57402258 IC50 = 9 nM T68782 CDJK52 57403006 IC50 = 150 nM T68782 CYG57I 57403305 IC50 = 32 nM T68782 CI68RM 57403987 IC50 = 50 nM T68782 CK76CI 57403988 IC50 = 14 nM T68782 CX13SU 57404015 IC50 = 85 nM T68782 C37SMZ 57505249 IC50 = 16000 nM T68782 C5KZ9N 59644708 IC50 > 10000 nM T68782 CX4V3U 59864915 IC50 = 350 nM T68782 C2D7LR 66967770 IC50 = 17 nM T68782 C0WK1P 67242411 IC50 = 82 nM T68782 CVM9Q1 68503758 IC50 > 10000 nM T68782 CA15ND 68505312 IC50 = 120 nM T68782 C0US2T 68505327 IC50 = 690 nM T68782 CX8W7F 68508048 IC50 = 2700 nM T68782 COJ4Q1 69315206 IC50 > 10000 nM T68782 CJ5Z7T 69316129 IC50 > 10000 nM T68782 CHX52Y 69561043 IC50 = 2 nM T68782 C6TB1K 70689410 IC50 > 10000 nM T68782 C6BFC9 70689411 IC50 > 10000 nM T68782 C0DC1J 70691517 IC50 > 10000 nM T68782 CTP4W6 70693611 IC50 > 10000 nM T68782 C40EGX 70693612 IC50 > 10000 nM T68782 CN42UV 70695720 IC50 > 10000 nM T68782 CAGV62 70695721 IC50 > 10000 nM T68782 C8XJ0I 71733818 IC50 = 4100 nM T68782 CXC78L 71733909 IC50 = 2200 nM T68782 C7B5XE 71733910 IC50 = 310 nM T68782 CQ21ZD 71733911 IC50 > 10000 nM T68782 CZG0S2 71733912 IC50 > 10000 nM T68782 CGBQ38 90479860 IC50 = 17 nM T68782 CKD3U1 90644206 IC50 = 45 nM T68782 CGP87O 90644207 IC50 = 9 nM T68782 CK13SY 90644208 IC50 = 62 nM T68782 CJNR26 90644209 IC50 = 8400 nM T68782 CLZJ36 118727285 EC50 = 21 nM T68782 CXWZ41 118727287 EC50 = 17 nM T68782 CL4AI3 118727288 EC50 = 25 nM T68782 CMDL48 118727289 EC50 = 44 nM T68782 C6X5EG 118727290 EC50 = 61 nM T68782 CB3QD7 118727291 EC50 = 6 nM T68782 CGFH47 118727294 EC50 = 1.7 nM T68782 CF6I8O 118727297 EC50 = 31 nM T68782 CE9G2Y 118727298 EC50 = 3 nM T68782 CCG76Q 118727299 EC50 = 11 nM T68782 CK9BJ0 118727300 EC50 = 24 nM T68782 CGAB46 118727301 EC50 = 180 nM T68782 CBN3D0 118727302 EC50 = 48 nM T68782 CVG17M 118727303 EC50 = 88 nM T68782 CZNC59 118727306 EC50 = 31 nM T68782 C8HZ9I 118727307 EC50 = 36 nM T68782 C3IXH8 118727308 EC50 = 40 nM T68782 CEK5C9 118727314 EC50 = 42 nM T68782 C3L5VY 118727315 EC50 = 48 nM T68782 C9M4YO 118727316 EC50 = 21 nM T68782 C4D5TR 134823954 Ki = 674 nM T68782 C6K7AM 135509970 IC50 = 16.98 nM T68782 CE79SV 138377584 IC50 = 3000 nM T68782 CU2C0Y 145968972 IC50 = 38 nM T68782 C8GDY6 145969532 IC50 = 13 nM T68782 CP6QG9 145970031 IC50 = 124 nM T68782 CG7BR1 145987034 Ki = 873 nM T68782 D01AFV 11500603 Ki = 5900 nM T68782 D02MXT 24952929 Ki > 3900 nM T68782 D03OYD 5311240 IC50 > 10000 nM T68782 D05GWV 11586961 Ki > 10000 nM T68782 D05HPB 11587023 Ki > 10000 nM T68782 D06HPV 10216733 Ki = 0.57 nM T68782 D07GCA 11514705 Ki = 1880 nM T68782 D07UDT 15551229 Ki > 500 nM T68782 D08CLB 346737 Ki > 10000 nM T68782 D08KZJ 11384493 Ki = 653 nM T68782 D0C0FU 43091550 Ki = 8900 nM T68782 D0E0HT 248828 Ki = 4740 nM T68782 D0I8MN 44441193 Ki = 4800 nM T68782 D0J5OX 16775011 Ki > 10000 nM T68782 D0J9PG 119461 Ki = 1400 nM T68782 D0O9ES 5311053 IC50 > 10000 nM T68782 D0QH5C 230826 Ki = 7600 nM T68782 D0S0BK 44441192 Ki > 10000 nM T68782 D0S2LO 9864831 Ki > 13000 nM T68782 D0TA0L 23685469 Ki > 1000 nM T68782 D0U5PC 43169594 Ki > 10000 nM T68782 D0Y1IF 23664784 Ki > 1000 nM T68782 D0Y4UG 44441190 Ki > 10000 nM T68782 D0Z3XJ 9817405 Ki > 500 nM T41145 CL80QG 11820 IC50 = 4800 nM T41145 C0NP2Q 351421 IC50 > 400000 nM T41145 CG5O0H 638578 IC50 = 53800 nM T41145 CZ3Y9X 2972356 IC50 = 330 nM T41145 CV9W7S 2988057 IC50 = 3162.28 nM T41145 C42AQR 4102773 IC50 > 14500 nM T41145 CT8G2Z 6458480 IC50 = 2511.89 nM T41145 C7EI6P 11745122 IC50 = 2100 nM T41145 CO3IL6 15990226 IC50 = 316.23 nM T41145 CZ91JF 15990296 IC50 = 125.89 nM T41145 C3SC0O 16026457 IC50 = 1900 nM T41145 CID57R 16026459 IC50 = 2000 nM T41145 CDB9H4 16026765 IC50 = 27000 nM T41145 CVW2J8 17568039 IC50 > 10000 nM T41145 C9R8UB 20895711 IC50 > 200000 nM T41145 CBO0Q4 20944521 IC50 = 3600 nM T41145 CWN9T6 20944522 IC50 = 3400 nM T41145 C3WP1E 20944528 IC50 = 5400 nM T41145 CE6HP0 20946705 IC50 = 1700 nM T41145 CN1IX5 20946712 IC50 = 4400 nM T41145 CG9NM2 20946713 IC50 = 3400 nM T41145 C60VPS 20946716 IC50 = 10500 nM T41145 C1ER4H 20946724 IC50 = 8700 nM T41145 C4MG9Q 20946727 IC50 = 11000 nM T41145 C4I2NX 20946734 IC50 = 794.33 nM T41145 C3M1XV 20969948 IC50 > 200000 nM T41145 C9YPE8 22110019 IC50 > 50000 nM T41145 C12TZA 22432992 IC50 = 630.96 nM T41145 CXL15A 22433053 IC50 = 398.11 nM T41145 CS1NE4 22433281 IC50 > 10000 nM T41145 CLJ74N 23609425 IC50 = 218000 nM T41145 COWB96 24489494 IC50 > 10000 nM T41145 C05CKD 24516170 IC50 > 10000 nM T41145 CIBE92 24789797 IC50 = 630.96 nM T41145 COB70I 24789844 IC50 = 316.23 nM T41145 C2JIY3 24790912 IC50 = 100 nM T41145 CZHU85 25330299 IC50 > 10000 nM T41145 C6YFX9 27331320 IC50 > 100000 nM T41145 CMSY09 27853996 IC50 > 100000 nM T41145 CN0J2C 29180108 IC50 = 100 nM T41145 CL1TP3 31954457 IC50 > 10000 nM T41145 C7GQ4B 32034429 IC50 > 10000 nM T41145 CV10FU 32318812 IC50 > 10000 nM T41145 CYGO57 42923164 IC50 > 50000 nM T41145 CG90JZ 42924396 IC50 > 10000 nM T41145 CN1I3A 42929656 IC50 = 195000 nM T41145 C06LRW 45873746 IC50 > 25000 nM T41145 C0PLT1 45873751 IC50 > 100000 nM T41145 CK3NP1 46249107 IC50 = 3162.28 nM T41145 C5HXW9 46249116 IC50 = 1584.89 nM T41145 CD06LA 46249215 IC50 = 125.89 nM T41145 CL31ZG 46339191 IC50 = 10100 nM T41145 CW4N5V 47035502 IC50 > 50000 nM T41145 C1QLE7 47046086 IC50 > 500000 nM T41145 CTU52G 49190366 IC50 = 590 nM T41145 CM6Y4O 49190451 IC50 = 420 nM T41145 CIS4D7 49190466 IC50 = 290 nM T41145 C2O3LN 50792180 IC50 > 200000 nM T41145 CVK20S 50792211 IC50 = 770 nM T41145 C37YMW 50792226 IC50 = 4400 nM T41145 CMJ7D0 50793116 IC50 = 22300 nM T41145 CDQ80N 50796602 IC50 = 660 nM T41145 CYP58I 50796734 IC50 = 270 nM T41145 CX12UC 50796762 IC50 = 290 nM T41145 C2GP8Q 50796763 IC50 = 3100 nM T41145 C5UQ8O 50796790 IC50 = 340 nM T41145 CP1U8X 50796792 IC50 = 680 nM T41145 C1R7BG 50796818 IC50 = 6720 nM T41145 CT34KZ 50796842 IC50 = 1170 nM T41145 CTSH48 50796873 IC50 = 790 nM T41145 CA01UQ 50796897 IC50 = 1050 nM T41145 CPZ93K 50820616 IC50 = 2240 nM T41145 CA2MT4 50820637 IC50 = 660 nM T41145 CVG1Y0 50820716 IC50 = 510 nM T41145 CKZH89 51043963 IC50 > 200000 nM T41145 CG3PR6 52912222 IC50 > 3.981 nM T41145 C76ZPW 71271926 IC50 = 9 nM T41145 CQOV07 75375570 IC50 = 30600 nM T41145 CJ47ZL 75435928 IC50 > 500000 nM T41145 CPY97E 83636605 IC50 = 190 nM T41145 C1Q9TW 86776557 IC50 = 240000 nM T41145 C9WB3G 95828281 IC50 > 20000 nM T41145 CZY31K 118721304 IC50 = 630.96 nM T41145 CYGS87 118721305 IC50 = 19952.62 nM T41145 CK16DC 118918689 IC50 = 93 nM T41145 COME25 118918694 IC50 = 910 nM T41145 CI6M3U 118918698 IC50 = 1200 nM T41145 C4T3AX 118918703 IC50 = 180 nM T41145 CF9J8E 118918705 IC50 = 12 nM T41145 C5GFE8 118918710 IC50 = 2200 nM T41145 CA3Z8O 118918714 IC50 = 43 nM T41145 CEM4Y1 118918717 IC50 = 520 nM T41145 CEJT45 118918718 IC50 = 1000 nM T41145 C3AZ9D 118918719 IC50 = 380 nM T41145 C8GLJ3 118918720 IC50 = 62 nM T41145 C8QA2X 118918735 IC50 = 15 nM T41145 CL27BG 118918739 IC50 = 1100 nM T41145 CAZR96 118918740 IC50 = 12 nM T41145 CBU9H2 118918747 IC50 = 39 nM T41145 C3AK9L 118918749 IC50 = 55 nM T41145 C0KI9P 118918753 IC50 = 52 nM T41145 C37ZJX 118932971 IC50 = 44 nM T41145 C4DF6I 118932972 IC50 = 56 nM T41145 C2ZY3U 118932975 IC50 = 53 nM T41145 C2O0NE 118932978 IC50 = 430 nM T41145 CHCU32 118932979 IC50 = 29 nM T41145 C2JCY3 118932989 IC50 = 100 nM T41145 CC14FI 118933132 IC50 = 7.9 nM T41145 CEPT12 118933133 IC50 = 15 nM T41145 CKY8H3 118933134 IC50 = 17 nM T41145 CGO91Y 118933136 IC50 = 60 nM T41145 CC35IE 118933137 IC50 = 24 nM T41145 C8AZ4C 119081691 IC50 > 20000 nM T41145 CUWX94 119081692 IC50 = 1500 nM T41145 CBD7I6 121232405 IC50 = 2.512 nM T41145 CM8UD0 121232406 IC50 = 1000 nM T41145 C3GD2W 121335190 IC50 > 20000 nM T41145 CECP26 121335281 IC50 > 20000 nM T41145 CDH8M4 121373418 IC50 > 20000 nM T41145 C47QXT 121376807 IC50 > 20000 nM T41145 CD3AR0 121559065 IC50 = 515000 nM T41145 CS9ZI3 122149386 IC50 = 293000 nM T41145 CWJD15 122705990 IC50 = 3150 nM T41145 CM8EB4 126961333 IC50 = 1550 nM T41145 CZ8S4U 127025422 IC50 = 310 nM T41145 CB3RH7 127025423 IC50 = 1400 nM T41145 C6TY8H 127025698 IC50 = 270 nM T41145 CTX9Y6 127029368 IC50 = 430 nM T41145 CT93VU 127029369 IC50 = 430 nM T41145 CFH9G7 127029370 IC50 = 2680 nM T41145 CV07YO 127038801 IC50 <= 1000 nM T41145 C4RGQ7 127043287 IC50 = 794.33 nM T41145 CF3Z9G 127043292 IC50 = 79.43 nM T41145 C3V9AN 127043657 IC50 = 316.23 nM T41145 CA3VI9 127043861 IC50 = 63.1 nM T41145 CCSJ69 127043862 IC50 = 1258.93 nM T41145 CJT6N0 127043863 IC50 = 125.89 nM T41145 CEG46M 127043864 IC50 = 31.62 nM T41145 CL8S6X 127043872 IC50 = 3162.28 nM T41145 CEAN18 127043873 IC50 = 1258.93 nM T41145 CZP0D9 127043874 IC50 = 5.012 nM T41145 C7Y1IB 127043875 IC50 = 15.85 nM T41145 CH4BE8 127043876 IC50 = 125.89 nM T41145 CWP65X 127043881 IC50 = 125.89 nM T41145 CO62HW 127044040 IC50 = 100 nM T41145 CE0CG1 127044041 IC50 = 1995.26 nM T41145 CCJ2T9 127044045 IC50 = 1258.93 nM T41145 CJ7YT3 127044046 IC50 = 79.43 nM T41145 CB5T0O 127044330 IC50 = 100 nM T41145 CYEW07 127044331 IC50 = 316.23 nM T41145 CAN9K0 127044332 IC50 = 1000 nM T41145 CH1MJ8 127044333 IC50 = 1258.93 nM T41145 CP15DV 127044334 IC50 = 794.33 nM T41145 CU7X9E 127044335 IC50 = 1584.89 nM T41145 CXN63Y 127044336 IC50 = 501.19 nM T41145 CLN5S3 127044787 IC50 = 199.53 nM T41145 CX4M3R 127044824 IC50 = 31.62 nM T41145 C5B9XC 127044825 IC50 = 125.89 nM T41145 CTY65A 127044826 IC50 = 100 nM T41145 C8F9IH 127044827 IC50 = 158.49 nM T41145 C0SOM8 127044828 IC50 = 100 nM T41145 CZ5H7K 127045294 IC50 = 50.12 nM T41145 CQOL84 127045572 IC50 = 1584.89 nM T41145 C2O9EX 127050976 IC50 = 650 nM T41145 C7NEB1 130471695 IC50 = 1150 nM T41145 CLA09E 130471696 IC50 = 1900 nM T41145 CWNY27 130471723 IC50 = 4150 nM T41145 CXW1B4 130471724 IC50 = 1010 nM T41145 C1EN7A 130471730 IC50 = 14200 nM T41145 C2HD6P 130471733 IC50 = 13300 nM T41145 C5DFI7 130471761 IC50 = 578 nM T41145 CDLE96 130471765 IC50 = 855 nM T41145 C1C8OB 130471770 IC50 = 591 nM T41145 CDC32I 130471775 IC50 = 3690 nM T41145 C3D7HE 130471777 IC50 = 2230 nM T41145 CFI30C 130471784 IC50 = 1310 nM T41145 C7TJA6 130471785 IC50 = 3310 nM T41145 CDUX50 130471789 IC50 = 1220 nM T41145 C8VAM6 130471790 IC50 = 1270 nM T41145 CN80UV 130471849 IC50 = 185 nM T41145 CEV5I3 130471855 IC50 = 547 nM T41145 CE1K3M 130471876 IC50 = 2300 nM T41145 CFTG42 130472058 IC50 = 5510 nM T41145 C5P2ED 130472268 IC50 = 4820 nM T41145 C7B6CZ 130472269 IC50 = 4540 nM T41145 CED70X 130472274 IC50 > 20000 nM T41145 CK0B6N 131985884 IC50 = 65 nM T41145 CGDN94 132275066 IC50 = 4600 nM T41145 CFXE14 137321203 IC50 > 100000 nM T41145 CXN4U1 137321204 IC50 = 19952.62 nM T41145 CPWF20 137632687 IC50 = 250 nM T41145 CD4NE1 137633137 IC50 = 170 nM T41145 CQT3A9 137636309 IC50 > 100000 nM T41145 CH07BA 137636753 IC50 = 110 nM T41145 CCAP49 137636933 IC50 = 630 nM T41145 CV1EP8 137639742 IC50 = 1000 nM T41145 CVC65R 137643133 IC50 = 160 nM T41145 CC3VL8 137644086 IC50 = 870 nM T41145 CC34KQ 137650533 IC50 = 220 nM T41145 CQ6XB7 139030526 IC50 > 100000 nM T41145 CD6U7X 145925666 IC50 = 567.5 nM T41145 CDI56Z 145982091 IC50 = 23600 nM T41145 CH4RJ3 145989398 IC50 > 200000 nM T41145 C0CFI1 145994298 IC50 = 16000 nM T41145 D03BTJ 15990224 IC50 = 79.43 nM T41145 D08RDI 35397514 IC50 = 270 nM T41145 D09ZPM 1091852 IC50 = 10000 nM T41145 D0C2PD 50796983 IC50 = 340 nM T41145 D0J6XI 1253361 IC50 = 199.53 nM T41145 D0O6XT 91827373 IC50 = 3.1 nM T41145 D0Q7IU 40642506 IC50 = 50.12 nM T99582 CY9A0M 66065 IC50 = 208 nM T99582 CWMH72 54768028 IC50 = 18900 nM T99582 C9DGW0 54768030 IC50 = 5800 nM T99582 C9VEX8 137656890 IC50 = 20500 nM T93662 D03SLR 445858 IC50 > 2000000 nM T93662 C73QJG 46210731 IC50 = 255000 nM T93662 C7US8R 46210732 IC50 = 102000 nM T93662 C67URQ 46210733 IC50 = 173000 nM T93662 C71KDG 46210734 IC50 = 120000 nM T93662 D04EWW 736186 IC50 > 2000000 nM T93662 D05PTT 5281792 IC50 = 545000 nM T93662 D0V9EN 689043 IC50 > 2000000 nM T36121 D0U3EP 445154 IC50 = 60000 nM T36121 C1B3ZR 2836600 IC50 = 146000 nM T36121 C42ENO 2836606 IC50 = 33000 nM T36121 CO8Y1R 5990469 IC50 = 29000 nM T36121 CBNH48 46898027 IC50 = 60000 nM T36121 CWVU38 85855478 IC50 = 1000 nM T36121 CPQ28F 86282373 IC50 = 34800 nM T36121 CF5X4H 118153396 IC50 = 3000 nM T36121 CX9Q7U 145982633 IC50 > 100000 nM T36121 CF73BG 145982638 IC50 = 7000 nM T36121 C3S9WQ 145982841 IC50 = 10000 nM T36121 C4D9RG 145983013 IC50 > 100000 nM T36121 CQ7M3D 145983111 IC50 = 30000 nM T36121 CB4SD3 145983842 IC50 > 100000 nM T36121 C71SMY 145984219 IC50 = 5000 nM T36121 C8U3PN 145984250 IC50 > 100000 nM T36121 CJID45 145984773 IC50 = 40000 nM T36121 CIC4Q0 145984776 IC50 = 40000 nM T36121 C03KHN 145984862 IC50 > 100000 nM T36121 CWK47Z 145985021 IC50 = 10000 nM T36121 C3QH1W 145985420 IC50 = 2500 nM T36121 C4BLP5 145985805 IC50 = 5000 nM T36121 C5YM1K 145985926 IC50 > 100000 nM T36121 CV9WN4 145986197 IC50 = 2000 nM T47888 D07UHS 107970 EC50 > 10000 nM T47888 D07UGA 5283560 IC50 = 0.23 nM T47888 D0I2RB 11502996 Ki > 5450 nM T47888 D0L9KH 44623998 EC50 > 10000 nM T47888 D0K4BI 10223146 IC50 = 10 nM T47888 D0PW0R 71547555 IC50 = 6.2 nM T47888 D0T8FV 23071856 IC50 = 1200 nM T47888 CPO6B9 2740144 IC50 > 10000 nM T47888 C7N5UR 4107292 IC50 > 10000 nM T47888 C89ATE 5309153 EC50 > 50000 nM T47888 C72DNW 9796603 IC50 = 86 nM T47888 CS8MB9 9821227 EC50 = 2107 nM T47888 C1K9GW 9824415 IC50 = 6500 nM T47888 CW37CN 9969355 EC50 > 10000 nM T47888 C7FGR9 9979368 IC50 > 10000 nM T47888 CZLT30 10045980 IC50 > 10000 nM T47888 CA4HX3 10125861 IC50 = 830 nM T47888 C8KXE2 10125862 IC50 = 99 nM T47888 CG6O1W 10125882 IC50 = 57 nM T47888 C7B8UT 10126584 IC50 = 1.7 nM T47888 CG65LQ 10126736 IC50 = 12 nM T47888 CN8H2S 10127475 IC50 > 10000 nM T47888 CCG97S 10127776 IC50 = 10 nM T47888 CGCK28 10149985 IC50 = 5.5 nM T47888 CO06YT 10150171 IC50 = 1.8 nM T47888 C3LG4R 10150372 IC50 = 1.8 nM T47888 CPU38H 10151146 IC50 = 1 nM T47888 CE9WX6 10172338 IC50 = 100 nM T47888 CDE1S4 10172354 IC50 = 6.3 nM T47888 CI5X6K 10172513 IC50 = 4 nM T47888 CWJO04 10172546 IC50 = 840 nM T47888 CS62VA 10173002 IC50 = 19 nM T47888 CL2QV0 10173327 IC50 = 8 nM T47888 CSV6Q3 10174181 IC50 = 3.9 nM T47888 C5XFN7 10174255 IC50 > 10000 nM T47888 C8XZV1 10174548 IC50 = 1.9 nM T47888 CG3DX8 10193676 IC50 = 200 nM T47888 CR9YM8 10193915 IC50 = 2 nM T47888 C5HJB9 10195325 IC50 > 10000 nM T47888 CY1T7W 10215138 IC50 = 86 nM T47888 C56XBS 10215741 IC50 = 680 nM T47888 CN2FJ9 10216035 IC50 = 1500 nM T47888 C6NP8S 10217498 IC50 > 10000 nM T47888 C9KH2F 10236683 IC50 = 200 nM T47888 CN93ZD 10249887 IC50 > 10000 nM T47888 C6H9VI 10249979 IC50 > 10000 nM T47888 C2O4UR 10251062 IC50 > 10000 nM T47888 C2YZC3 10271422 IC50 = 230 nM T47888 CN0EC2 10286857 IC50 = 60 nM T47888 CKPV49 10287091 IC50 = 110 nM T47888 C74CKG 10287343 IC50 = 24 nM T47888 CW5JG7 10287365 IC50 = 2.6 nM T47888 C3R1AI 10288370 IC50 = 6.1 nM T47888 C5MDF6 10288527 IC50 > 10000 nM T47888 C6EY2U 10289318 IC50 = 3 nM T47888 CJ26CW 10308738 IC50 = 66 nM T47888 C2U3LT 10309022 IC50 = 4400 nM T47888 C8VP3G 10309271 IC50 = 41 nM T47888 C7B2FU 10309462 IC50 = 0.8 nM T47888 CAF85E 10310253 IC50 = 2.9 nM T47888 CPK61C 10310952 IC50 > 10000 nM T47888 C8HBY4 10311227 IC50 = 1.5 nM T47888 C3SM5Z 10317453 IC50 > 10000 nM T47888 CG89DO 10363915 IC50 > 10000 nM T47888 CDV3W7 10384596 IC50 = 4.5 nM T47888 C8WL6R 10408874 IC50 > 10000 nM T47888 COQ65E 10409838 IC50 > 10000 nM T47888 CI3EW1 10430549 IC50 > 10000 nM T47888 CAL72D 10476387 IC50 > 10000 nM T47888 C9NRD6 11168252 IC50 > 10000 nM T47888 CD8T1W 11222939 EC50 > 5000 nM T47888 CUR1P8 11224984 EC50 > 10000 nM T47888 CFPH94 11248292 IC50 > 10000 nM T47888 CK65MP 11271470 IC50 > 10000 nM T47888 CYH0U8 11408903 IC50 > 10000 nM T47888 CER35T 11466640 IC50 > 10000 nM T47888 CW51YT 11495139 IC50 > 10000 nM T47888 CDE78J 11496072 IC50 > 10000 nM T47888 C7EOU1 11501764 IC50 > 10000 nM T47888 CR1ME9 11501873 EC50 > 10000 nM T47888 CS27OX 11502026 IC50 > 10000 nM T47888 CVW6Q3 11575787 IC50 > 10000 nM T47888 CB75ZP 11575913 EC50 > 10000 nM T47888 CXS54Q 11603220 IC50 > 10000 nM T47888 CCW90K 11603726 EC50 > 10000 nM T47888 C96LNP 11604577 IC50 > 10000 nM T47888 CAN4Q9 11611053 EC50 > 10000 nM T47888 C41XAE 11624780 EC50 > 10000 nM T47888 CCY7J2 11626664 EC50 > 10000 nM T47888 CA8W5N 11646599 EC50 > 10000 nM T47888 CYS5F1 11653967 IC50 > 10000 nM T47888 CMJ32O 11662328 IC50 > 10000 nM T47888 CVG41H 11682696 EC50 > 10000 nM T47888 CCF80W 11689680 EC50 > 10000 nM T47888 C0BR1U 11696807 IC50 > 10000 nM T47888 CK5S1L 11697013 EC50 > 10000 nM T47888 C4G2OP 11743459 IC50 > 10000 nM T47888 CZ6YN9 11752659 IC50 > 10000 nM T47888 CDI32A 16038017 EC50 > 10000 nM T47888 CGAD08 17253208 EC50 > 50000 nM T47888 CIEK03 17253281 EC50 > 50000 nM T47888 C6HB9A 21455530 IC50 = 12 nM T47888 CL41AD 23071887 IC50 = 2800 nM T47888 C8WYV6 23071917 IC50 = 3900 nM T47888 CTLG80 23071955 IC50 = 9500 nM T47888 C6N8QR 23071977 IC50 = 1600 nM T47888 CY3GD5 23072004 IC50 = 2200 nM T47888 CWA4P5 23072092 IC50 = 1200 nM T47888 C5ETR1 23072144 IC50 = 1200 nM T47888 C6I0ED 24812110 IC50 = 0.8 nM T47888 C0O9UG 24825338 EC50 > 10000 nM T47888 CB82GW 24825339 IC50 > 10000 nM T47888 C14EAK 25110484 EC50 > 50000 nM T47888 C01FRW 25110488 EC50 > 50000 nM T47888 CXU68J 25110496 EC50 > 50000 nM T47888 CI2VH9 25110498 EC50 > 50000 nM T47888 CLEF36 25110499 EC50 > 50000 nM T47888 C10HKX 25192001 EC50 > 5000 nM T47888 C48TPJ 42630194 EC50 > 100000 nM T47888 CDL1C8 44125170 EC50 > 33113.11 nM T47888 CG73ST 44138103 EC50 > 100000 nM T47888 CH8CM7 44341291 IC50 = 73 nM T47888 CQR2G1 44341399 IC50 = 76 nM T47888 C8NOT7 44342221 EC50 = 973.2 nM T47888 CCN68O 44342231 EC50 > 5000 nM T47888 CXJ08Y 44342244 EC50 = 2685 nM T47888 C6LT8S 44342246 EC50 = 2760 nM T47888 CMKZ19 44344194 IC50 = 150 nM T47888 CLQ25X 44344210 IC50 = 19 nM T47888 C31BXA 44344270 IC50 = 1.8 nM T47888 CY7FC4 44344298 IC50 = 1.4 nM T47888 C1SP9M 44344338 IC50 = 2000 nM T47888 C2D5LZ 44344360 IC50 = 140 nM T47888 CT4NW0 44344390 IC50 = 530 nM T47888 C9S2FH 44344404 IC50 = 11 nM T47888 CY9C1D 44344412 IC50 = 2200 nM T47888 CLDU29 44344413 IC50 = 45 nM T47888 C91OKY 44344446 IC50 = 450 nM T47888 CL3CT8 44344456 IC50 = 110 nM T47888 CJ36UD 44394116 IC50 = 2200 nM T47888 C5KA6D 44394117 IC50 > 1000 nM T47888 CU7L0K 44394153 IC50 > 1000 nM T47888 CT8UN6 44394161 IC50 > 1000 nM T47888 C9E6CF 44394169 IC50 > 1000 nM T47888 C8H0XM 44394191 IC50 = 422 nM T47888 CH2A5S 44394211 IC50 > 1000 nM T47888 CND39O 44394212 IC50 = 760 nM T47888 C84JPI 44394247 IC50 > 1000 nM T47888 CA28OJ 44394273 IC50 > 1000 nM T47888 CO0T1E 44394279 IC50 = 330 nM T47888 CL5BC6 44394330 IC50 > 1000 nM T47888 C4DIT3 44398076 EC50 = 18 nM T47888 CDY46P 44412165 IC50 > 10000 nM T47888 CR2DT4 44412221 IC50 > 10000 nM T47888 CRV34X 44412232 IC50 > 10000 nM T47888 CV63YC 44412233 IC50 > 10000 nM T47888 CQ1V3J 44412282 IC50 > 10000 nM T47888 CB6KR7 44412294 IC50 > 10000 nM T47888 CTV5M0 44412353 IC50 > 10000 nM T47888 CN7K2O 44412364 IC50 > 10000 nM T47888 CL1GJ3 44412415 IC50 > 10000 nM T47888 CV28IK 44412416 IC50 > 10000 nM T47888 CBM50W 44412428 IC50 > 10000 nM T47888 C05TUB 44412658 EC50 > 10000 nM T47888 CH51GD 44412659 EC50 > 10000 nM T47888 C3M5SO 44412702 EC50 > 10000 nM T47888 CBUQ92 44412827 EC50 > 10000 nM T47888 CM8IK4 44412854 EC50 > 10000 nM T47888 CBL87K 44412867 EC50 > 10000 nM T47888 COA6Q1 44412868 EC50 > 10000 nM T47888 C80JSN 44412882 EC50 > 10000 nM T47888 C2WV6S 44412883 EC50 > 10000 nM T47888 C84PLZ 44412908 EC50 > 10000 nM T47888 C78DOK 44412936 EC50 > 10000 nM T47888 CH6Z8V 44412962 EC50 > 10000 nM T47888 C3MWD4 44412971 EC50 > 10000 nM T47888 CJC06H 44412994 EC50 > 10000 nM T47888 CT6EU7 44413274 IC50 > 10000 nM T47888 CYO6R3 44413349 IC50 > 10000 nM T47888 CH9NL4 44413365 IC50 > 10000 nM T47888 CW8E0R 44413415 IC50 > 10000 nM T47888 CYW5D3 44413430 IC50 > 10000 nM T47888 CJ5S2H 44413446 IC50 > 10000 nM T47888 CWRZ40 44413447 IC50 > 10000 nM T47888 CVC61G 44413482 IC50 > 10000 nM T47888 C0I3LB 44422601 EC50 = 270 nM T47888 C2O7AP 44422604 EC50 = 490 nM T47888 C7O0PC 44422606 EC50 = 530 nM T47888 C2WEQ7 44437392 IC50 = 24000 nM T47888 CP1FN6 44437417 IC50 = 11000 nM T47888 C0W3FQ 44439850 IC50 > 10000 nM T47888 CB4Z3I 44439851 IC50 > 10000 nM T47888 C9SFT8 44439852 IC50 > 10000 nM T47888 CS9H0L 44517795 EC50 > 100000 nM T47888 CX13MK 44547414 EC50 > 100000 nM T47888 CYOW10 45377016 IC50 > 10000 nM T47888 C7D3LB 45377018 IC50 > 10000 nM T47888 CN0A4O 45377161 IC50 > 10000 nM T47888 C8ELI4 45378010 IC50 > 10000 nM T47888 C73DCB 46174905 EC50 > 10000 nM T47888 CPU02J 46190696 IC50 > 10000 nM T47888 CQY5P8 46866185 IC50 > 22000 nM T47888 C6LJ7A 46866186 IC50 > 22000 nM T47888 CW6RX2 46881847 IC50 > 22000 nM T47888 CE32QB 46881848 IC50 > 22000 nM T47888 CAHC81 46881875 IC50 > 22000 nM T47888 C0BOR7 46881876 IC50 > 22000 nM T47888 CCS12Z 46881877 IC50 > 22000 nM T47888 C3QMS1 46881912 IC50 > 22000 nM T47888 CTL89X 46884020 EC50 > 5000 nM T47888 C5Z6RM 49839234 EC50 = 10000 nM T47888 C4BXP1 49848557 EC50 > 31622.78 nM T47888 CD2MT6 51000470 IC50 = 3000 nM T47888 C1DYT0 53358422 IC50 = 3900 nM T47888 CC7DZ4 53362086 EC50 > 10000 nM T47888 CU3Y6D 53388307 IC50 = 1100 nM T47888 CE3M4W 54582606 IC50 = 2800 nM T47888 CWNO65 54582607 IC50 = 2800 nM T47888 C4M8ZE 54583567 IC50 = 2600 nM T47888 C8PKX0 54587490 IC50 = 2400 nM T47888 CU62DN 54764919 EC50 > 25000 nM T47888 CBIH06 56954024 IC50 > 10000 nM T47888 CKWG20 57390239 EC50 = 3650 nM T47888 C5YS7U 58329611 EC50 > 10000 nM T47888 C5UTG1 66829311 EC50 > 1000 nM T47888 CHZG64 67009121 IC50 > 10000 nM T47888 C6AZY0 67249162 EC50 > 10000 nM T47888 CX6SF2 67250226 EC50 > 10000 nM T47888 CY09OV 69263869 EC50 > 10000 nM T47888 CR4V0T 71450073 EC50 > 10000 nM T47888 C2P3UC 71547556 IC50 = 2.3 nM T47888 CJP7X1 71547558 IC50 = 5.2 nM T47888 CZ9FX8 71547628 IC50 = 12 nM T47888 CL3Y8J 89484779 IC50 = 3.7 nM T47888 CQ3PK4 90308914 IC50 = 21 nM T47888 CHLT53 90308956 IC50 = 3.6 nM T47888 C89FXZ 90309040 IC50 = 27 nM T47888 C72CPK 90309054 IC50 = 39 nM T47888 CVUB74 90309056 IC50 = 76 nM T47888 C63RDX 90309065 IC50 = 20 nM T47888 CR4J2L 90309098 IC50 = 21 nM T47888 CYSQ05 90309100 IC50 = 88 nM T47888 CH7VQ0 90309119 IC50 = 11 nM T47888 C8EH3B 90309141 IC50 = 8.8 nM T47888 CL74JM 90309142 IC50 = 8.2 nM T47888 C6QW5D 90309191 IC50 = 17 nM T47888 CVA62H 90309206 IC50 = 83 nM T47888 C9LSD1 90309218 IC50 = 29 nM T47888 CA01FL 90309243 IC50 = 9.3 nM T47888 CDO0Z3 90309325 IC50 = 4 nM T47888 CPHM13 90309435 IC50 = 17 nM T47888 CCZW83 90309510 IC50 = 39 nM T47888 CN9R6C 90309512 IC50 = 8.8 nM T47888 CY3ZT1 90309524 IC50 = 45 nM T47888 CMY54W 90343274 IC50 = 6.4 nM T47888 C50KHV 118727601 IC50 = 1300 nM T47888 CQ5P6A 118727602 IC50 = 21000 nM T47888 CCK80O 118727603 IC50 > 25000 nM T47888 C6SCL3 118728423 IC50 = 820 nM T47888 C5Q7NY 118728424 IC50 = 1500 nM T47888 C30WSN 118728425 IC50 = 500 nM T47888 C9OA7Y 118728426 IC50 = 860 nM T47888 C85AFZ 118728427 IC50 = 1400 nM T47888 CNI96W 118728428 IC50 = 980 nM T47888 C3O6KB 118728429 IC50 = 84 nM T47888 C4U3DG 118728430 IC50 = 13 nM T47888 C8U0GE 118728431 IC50 = 43 nM T47888 C72NCP 118728432 IC50 = 45 nM T47888 C2YHT8 118728433 IC50 = 210 nM T47888 C4M3YA 118728434 IC50 = 390 nM T47888 C1ZR2H 122190861 IC50 = 1100 nM T47888 CB57SG 122190862 IC50 > 25000 nM T47888 CC34ZI 122190863 IC50 > 25000 nM T47888 CCR6M9 122190864 IC50 = 123 nM T47888 C9U4QR 124221654 EC50 > 100000 nM T47888 C4O8CF 127027731 IC50 = 25 nM T47888 C64DPO 127029521 IC50 = 34 nM T47888 CUE0N7 134130169 EC50 > 100000 nM T47888 C3NC1O 134130546 EC50 > 100000 nM T47888 CJH4K9 134130548 EC50 > 100000 nM T47888 C6JB4Z 134130695 EC50 > 100000 nM T47888 C6V4DA 134130884 EC50 > 100000 nM T47888 CNVC46 134131381 EC50 > 100000 nM T47888 CR0Z3M 145964351 IC50 > 1000 nM T47888 CLX67W 145964960 IC50 > 1000 nM T47888 CTP5Q0 145965024 IC50 > 1000 nM T47888 CXGD49 145965534 IC50 > 1000 nM T47888 CF7CL1 145966048 IC50 > 1000 nM T47888 C0ZM4R 145966230 IC50 = 56.5 nM T47888 CNZI51 145966801 IC50 > 1000 nM T47888 CI83OB 145974612 IC50 > 1000 nM T47888 CY8IH7 145976116 IC50 > 1000 nM T47888 C6JW8K 145976329 IC50 = 29.1 nM T47888 COJ29A 145977506 IC50 > 1000 nM T47888 C9J4HN 155317213 IC50 > 1000 nM T47888 CZ76KV 155317216 IC50 > 1000 nM T47888 CPUQ19 155317219 IC50 > 1000 nM T47888 C2TB6V 155317220 IC50 = 270.3 nM T47888 CCHR02 155317224 IC50 > 1000 nM T47888 CE3W9F 155317227 IC50 = 188.5 nM T47888 C9XOY4 155317228 IC50 > 1000 nM T47888 CRF7V0 155317229 IC50 = 29.9 nM T47888 CN12PQ 155317230 IC50 = 278.5 nM T47888 CQ35OR 155317231 IC50 > 1000 nM T47888 C7X6US 155317234 IC50 > 1000 nM T47888 C5LNV9 155317237 IC50 > 1000 nM T47888 CJX1S6 155317240 IC50 > 1000 nM T47888 CTQC16 155317243 IC50 = 194.5 nM T47888 C9A7VF 155317245 IC50 > 1000 nM T47888 CG79DH 155317246 IC50 > 1000 nM T47888 C0BE9I 155317247 IC50 = 296.5 nM T47888 CVSC94 155317248 IC50 = 359.3 nM T47888 C2F4VY 155317251 IC50 > 1000 nM T47888 CZR01A 155317256 IC50 > 1000 nM T47888 CX76PB 155317261 IC50 = 38.5 nM T47888 CW10AC 155317265 IC50 = 14.6 nM T47888 C3ZO2T 155317271 IC50 > 1000 nM T47888 CZO3N6 155317275 IC50 = 362.3 nM T47888 C43CXP 155317276 IC50 = 66.7 nM T47888 CEHG92 155317278 IC50 > 1000 nM T47888 CLG86C 155317279 IC50 = 73.3 nM T47888 CJ6R9A 155317280 IC50 > 1000 nM T47888 D00VHN 46905530 IC50 = 1100 nM T47888 D02LTS 59393720 IC50 > 10000 nM T47888 D04IAF 11452022 IC50 = 5.9 nM T47888 D04XCB 10149595 IC50 = 3300 nM T47888 D06DYN 9908268 IC50 = 1100 nM T47888 D06XMB 44394220 IC50 > 1000 nM T47888 D07EAB 10215259 IC50 > 10000 nM T47888 D08VLT 10125714 IC50 = 1000 nM T47888 D0D5QS 11725751 IC50 = 0.7 nM T47888 D0LO4T 10287034 IC50 > 1000 nM T47888 D0N0BN 44394248 IC50 > 1000 nM T47888 D0P1TY 44344193 IC50 = 580 nM T47888 D0P2AZ 10149721 IC50 > 10000 nM T47888 D0ZU0O 4077460 IC50 > 10000 nM T98311 D00HDU 91270 IC50 = 2.6 nM T98311 D00SEB 5388962 IC50 = 1.2 nM T98311 D01FJT 656604 IC50 = 7244359.6 nM T98311 D01STB 5362129 IC50 = 4 nM T98311 D03KYG 107807 IC50 = 1.5 nM T98311 D07HGR 5362119 IC50 = 0.1 nM T98311 D0DZ3X 145742 Ki = 86000 nM T98311 D0E6XR 3062316 Ki = 715000 nM T98311 D0I0EG 44093 IC50 = 0.63 nM T98311 D0I7SZ 54892 IC50 = 8.3 nM T98311 D0M5OC 5484727 IC50 = 0.93 nM T98311 D0N5HJ 5462501 IC50 = 1.2 nM T98311 D0N6RF 65999 Ki = 6000 nM T98311 D0Q0PR 54675769 Ki = 167000 nM T98311 D0U2JP 4369359 IC50 = 11000 nM T98311 D0U3EC 5362124 IC50 = 1.7 nM T98311 D09JES 6324648 Ki = 13.8 nM T98311 D0N4IV 10718956 IC50 > 1000 nM T98311 D04MBS 9801007 IC50 = 12 nM T98311 D05NRI 189729 IC50 = 36.31 nM T98311 D05UQD 656629 Ki = 0.015 nM T98311 D06WBA 123742 IC50 = 32000 nM T98311 D0I5QZ 9998020 IC50 = 30 nM T98311 D0K9YR 9810328 IC50 = 2.5 nM T98311 D0T2IQ 443600 IC50 > 100000 nM T98311 CQP46K 3937 IC50 = 3.981 nM T98311 CSH72V 4802 IC50 = 5.012 nM T98311 CXY67D 11163 IC50 = 7244359.6 nM T98311 C43SDH 62956 Ki = 1.5 nM T98311 C7QUA0 71244 IC50 = 3.715 nM T98311 C2N6DR 71320 IC50 = 7 nM T98311 CAM5C0 73086 IC50 = 3801893.96 nM T98311 CZ0M7X 81721 IC50 = 309029.54 nM T98311 C5F9KD 83525 Ki = 50000 nM T98311 C19KSO 85362 IC50 = 10000 nM T98311 C49UDX 88079 IC50 = 1202264.43 nM T98311 C7KR0D 92181 IC50 = 30199.52 nM T98311 CIWS40 92400 IC50 = 0.4 nM T98311 CCOI47 92829 IC50 = 208929.61 nM T98311 CR71YD 92843 IC50 = 2511886.43 nM T98311 C7E9ND 92946 IC50 = 87096.36 nM T98311 C57WLO 92953 IC50 = 602559.59 nM T98311 C2TD8W 96814 IC50 = 190546.07 nM T98311 C3GQ5H 97054 IC50 = 5888436.55 nM T98311 CQL18W 97363 IC50 = 9120108.39 nM T98311 CY23QB 97364 IC50 = 8709635.9 nM T98311 CR01ON 99278 IC50 = 5370317.96 nM T98311 CRE70Y 99978 IC50 = 199.53 nM T98311 C4MKD1 101179 IC50 = 6309573.44 nM T98311 C0WN9F 107994 IC50 = 2.8 nM T98311 CJ1W2Z 108985 IC50 = 229086.77 nM T98311 CP5Q6B 111257 IC50 = 5754399.37 nM T98311 CTM7W0 114973 IC50 = 3.2 nM T98311 CM9S5Q 122113 IC50 = 19.95 nM T98311 CGR1J3 123913 IC50 = 7079457.84 nM T98311 CPIJ02 130842 IC50 = 9400 nM T98311 C0VK5M 133560 IC50 = 1000 nM T98311 CWPS82 133842 IC50 = 1000000000 nM T98311 CRB2Z1 134166 IC50 = 1 nM T98311 C6ZQJ0 137365 IC50 = 31.62 nM T98311 C6XMS5 150903 IC50 = 912010.84 nM T98311 CDCS28 150964 IC50 = 229086.77 nM T98311 C7CN8P 151148 IC50 = 14125375.45 nM T98311 CMY75U 151282 IC50 = 1412537.54 nM T98311 CB3D6T 156271 IC50 = 12 nM T98311 C6TDE7 165505 IC50 = 2818.38 nM T98311 CB9Q1L 168182 IC50 = 1584.89 nM T98311 CLJ9D1 189008 IC50 = 3235936.57 nM T98311 C0R3KO 194156 IC50 = 33113.11 nM T98311 CU0B8E 329113 IC50 = 1096478.2 nM T98311 CJX54Q 335542 IC50 = 10 nM T98311 CP2T7N 443376 IC50 = 220 nM T98311 CO1UK9 444876 IC50 = 128824.96 nM T98311 C9VSE5 446549 IC50 = 10964.78 nM T98311 CZGF79 448982 IC50 = 23 nM T98311 C1BTQ3 494324 IC50 = 12.59 nM T98311 CN67CR 555078 IC50 > 100000 nM T98311 CQ6IO0 1551643 IC50 = 1995262.31 nM T98311 C2AS3C 2724807 IC50 = 4570881.9 nM T98311 CSE85T 2828746 IC50 = 300 nM T98311 C79HSA 2828749 IC50 = 200000 nM T98311 CF47UW 2834684 IC50 = 20 nM T98311 CN52PM 3013625 IC50 = 446683.59 nM T98311 C8SU0O 3033702 IC50 = 0.8 nM T98311 CA6E1H 3080576 IC50 = 5370317.96 nM T98311 C7YDX5 3082827 IC50 = 0.2951 nM T98311 CY36MH 4369380 IC50 = 140 nM T98311 CH01XT 5281656 Ki = 250200 nM T98311 CO58XD 5311161 IC50 > 100000 nM T98311 CF8YR2 5464343 IC50 = 9900 nM T98311 C1YI9C 5464344 IC50 = 1.7 nM T98311 CMAH79 5479774 Ki = 34200 nM T98311 CJHI21 5484352 IC50 = 616595 nM T98311 CF49DL 5490790 Ki = 1.4 nM T98311 CH5U2F 5491963 IC50 = 3801893.96 nM T98311 CF07VG 5496455 IC50 = 457088.19 nM T98311 CTCZ08 5748613 IC50 = 730 nM T98311 C1QBP5 6426706 IC50 = 3235936.57 nM T98311 CV1E8W 6426709 IC50 = 16982436.52 nM T98311 CO03CU 6427013 IC50 = 10000000 nM T98311 C1A6GP 6427052 IC50 = 10000000 nM T98311 C7XIW1 6992396 IC50 = 190546.07 nM T98311 C9W1MN 6992506 IC50 = 10000000 nM T98311 CB5YC3 6992691 IC50 = 7413102.41 nM T98311 CQ5E0R 6992869 IC50 = 1202264.43 nM T98311 CY8UR9 6992873 IC50 = 128824.96 nM T98311 C8Z9OD 6992930 IC50 = 4786300.92 nM T98311 CWC8M3 6993111 IC50 = 1096478.2 nM T98311 CK3Q0Z 6993120 IC50 = 52480.75 nM T98311 C7HIQ9 6998029 IC50 = 2511886.43 nM T98311 CMB48H 7009555 IC50 = 21877.62 nM T98311 C4UO5E 7009596 IC50 = 933254.3 nM T98311 C46LAM 7009644 IC50 = 8511380.38 nM T98311 CH7P4I 7009653 IC50 = 15848.93 nM T98311 C15XOM 7010504 IC50 = 380189.4 nM T98311 C7QV9R 7019085 IC50 = 1995.26 nM T98311 CFW5P0 7020333 IC50 = 457088.19 nM T98311 CP4M1Q 7021854 IC50 = 1995262.31 nM T98311 C36DHQ 7022320 IC50 = 3235936.57 nM T98311 C2PR6I 7023107 IC50 = 3090295.43 nM T98311 CP0BE5 7039484 IC50 = 549540.87 nM T98311 C28NMU 7408195 IC50 = 3715.35 nM T98311 CPU01J 7408255 IC50 = 2300 nM T98311 C5Q9ZO 9601226 IC50 = 1 nM T98311 C02INA 9803222 IC50 = 140 nM T98311 CEX1W2 9822849 IC50 = 87 nM T98311 CDO9J0 9837272 IC50 = 416869.38 nM T98311 CRF51I 9839564 IC50 > 10000 nM T98311 CI7Q0Y 9840601 IC50 = 1400 nM T98311 CZ2HC0 9840687 IC50 = 175 nM T98311 C2MEU1 9844054 IC50 = 52 nM T98311 C38BVX 9870100 IC50 > 1000 nM T98311 C03SVH 9882882 IC50 = 18700 nM T98311 CZ20AN 9905282 IC50 = 12000 nM T98311 C1NDX9 9910508 IC50 = 10000 nM T98311 CVPG59 9932329 IC50 = 35 nM T98311 CVG0O2 9959014 IC50 > 1000 nM T98311 CU61CH 9978465 IC50 = 260 nM T98311 C91HDB 10014925 IC50 = 2300 nM T98311 C8SY5F 10015450 Ki = 126000 nM T98311 C5UH9J 10041763 IC50 = 4 nM T98311 CMD3J1 10047309 IC50 = 4.8 nM T98311 C32OGJ 10071569 IC50 = 25 nM T98311 CH93JG 10093438 IC50 = 460 nM T98311 C63CBL 10107034 IC50 = 11000 nM T98311 CG0DW7 10141595 IC50 > 100000 nM T98311 C05YBI 10336328 IC50 = 10000 nM T98311 CS3ND2 10355231 IC50 = 769000 nM T98311 C5D8ZA 10355232 Ki = 14200 nM T98311 CL73JY 10381547 IC50 = 5000 nM T98311 C4GZ8V 10393285 IC50 = 50 nM T98311 CM0S1U 10426368 IC50 = 16100 nM T98311 CX78MU 10432045 IC50 = 92 nM T98311 CS4G3H 10436816 IC50 > 100000 nM T98311 CU6OH3 10448308 IC50 = 34 nM T98311 CX38EB 10467565 IC50 = 90000 nM T98311 CG6FZ1 10475845 IC50 = 1.698 nM T98311 C9XC8Y 10493383 IC50 = 34000 nM T98311 C4VN0M 10494952 IC50 > 10000 nM T98311 C69RND 10496022 IC50 = 2000 nM T98311 CG32FM 10613145 IC50 > 100000 nM T98311 CQN7S4 10664538 IC50 = 725 nM T98311 C4S3EZ 10710922 IC50 = 1400 nM T98311 CI4SQ2 10732349 IC50 > 100000 nM T98311 CAD84L 10735551 IC50 > 10000 nM T98311 CT78AR 10759255 IC50 = 118 nM T98311 C7O6RU 10759256 IC50 > 10000 nM T98311 CLAP90 10785969 IC50 > 1000 nM T98311 CM74LH 10789594 IC50 > 1000 nM T98311 CFUE14 10829618 IC50 = 8000 nM T98311 C3UCL2 10854279 IC50 = 12400 nM T98311 CKAF49 10900068 IC50 > 1000 nM T98311 CV70TF 10900407 IC50 = 257039.58 nM T98311 CA7B4P 11119038 IC50 = 457.09 nM T98311 C8Q1SZ 11176510 IC50 = 600 nM T98311 CSF91W 11191083 IC50 = 3.8 nM T98311 CC0MU7 11192220 IC50 > 100000 nM T98311 C4ON0L 11442784 IC50 = 72 nM T98311 CE3HA6 11556698 Ki = 0.65 nM T98311 C78VRX 11774785 IC50 = 4000 nM T98311 COT0R7 11792153 IC50 = 22 nM T98311 CJ4VL3 11797382 IC50 > 1000 nM T98311 CSD43L 11989733 IC50 = 20000 nM T98311 C9IG0H 11992410 Ki = 195700 nM T98311 CJK95A 11992491 Ki = 84300 nM T98311 CTL5N6 11992492 Ki = 33600 nM T98311 CSK08P 11992493 Ki = 13300 nM T98311 C6YAP0 11992494 Ki = 43000 nM T98311 CG2ZY3 12190925 IC50 = 1348962.88 nM T98311 C57JAK 12698983 IC50 = 33000 nM T98311 CNU93T 12698984 IC50 = 3700 nM T98311 CRE7O9 12698990 IC50 = 35000 nM T98311 CPE6H9 12698991 IC50 = 30000 nM T98311 CQ6T3P 12698992 IC50 = 19000 nM T98311 C53CVG 12698999 IC50 = 100000 nM T98311 CW3DV9 12785186 IC50 = 67608.3 nM T98311 CC1GB9 12854254 IC50 = 70 nM T98311 CCXB83 12854279 IC50 = 86 nM T98311 C16NQY 12876150 IC50 = 19054.61 nM T98311 C0S2BY 12883918 IC50 = 130 nM T98311 CPV89D 12942866 IC50 = 18 nM T98311 C06PUC 12942868 IC50 = 19.95 nM T98311 CH6GO8 13036940 IC50 = 851.14 nM T98311 CL6T9B 13036944 IC50 = 426.58 nM T98311 C3B6JL 13036947 IC50 = 3019.95 nM T98311 CNU7I4 13044267 IC50 = 300 nM T98311 C58IDW 13044278 IC50 = 3 nM T98311 CGN26M 13069290 IC50 = 100 nM T98311 CDXC29 13104362 IC50 = 72.44 nM T98311 CG4MW9 13105154 IC50 = 1.202 nM T98311 CQT32M 13135337 IC50 = 39.81 nM T98311 CUOP05 13136851 IC50 = 12.59 nM T98311 C2CPA7 13136852 IC50 = 3.981 nM T98311 CCZY61 13144519 IC50 = 2511.89 nM T98311 C83XMT 13144525 IC50 = 1 nM T98311 CQ4DK3 13144530 IC50 = 3162.28 nM T98311 CY05BC 13144539 IC50 = 125.89 nM T98311 C6UFA7 13208321 IC50 = 38904.51 nM T98311 CC9Q7D 13241661 IC50 = 1.995 nM T98311 CD32WB 13335293 IC50 = 39.81 nM T98311 CUOH03 13339952 IC50 = 13 nM T98311 CY6G3M 13375125 IC50 = 3 nM T98311 C1X4KC 13456344 IC50 = 1.7 nM T98311 C3M7TP 13456346 IC50 = 2400 nM T98311 CB2MK0 13456353 IC50 = 5100 nM T98311 CNC8Z9 13456366 IC50 = 1.6 nM T98311 CBA7E6 13456368 IC50 = 2400 nM T98311 CP39OT 13456371 IC50 = 7900 nM T98311 CNW9U6 13456375 IC50 = 1.5 nM T98311 CHE38M 13456380 IC50 = 2.1 nM T98311 C3KAG2 13456384 IC50 = 3.3 nM T98311 CVKP79 13456389 IC50 = 11 nM T98311 CQN8H1 13456394 IC50 = 2.1 nM T98311 CE48FZ 13456399 IC50 = 2.4 nM T98311 CXDK27 13456404 IC50 = 2.3 nM T98311 CK49UY 13456423 IC50 = 6.7 nM T98311 C4TW5G 13477728 IC50 = 2200 nM T98311 C0U9VL 13500748 IC50 = 40 nM T98311 C1WZD8 13500752 IC50 = 15 nM T98311 CF0B3X 13500754 IC50 = 4 nM T98311 C2KD8I 13500765 IC50 = 2.9 nM T98311 C7WFB0 13500770 IC50 = 7 nM T98311 C20UNH 13500773 IC50 = 4 nM T98311 CJUH76 13500778 IC50 = 8.5 nM T98311 CZU08S 13500788 IC50 = 540 nM T98311 C9SL4H 13500790 IC50 = 45 nM T98311 C4VUX3 13500793 IC50 = 1000 nM T98311 CV4DT1 13500795 IC50 = 5 nM T98311 CE04SO 13500798 IC50 = 2600 nM T98311 CX4TI6 13500800 IC50 = 6.5 nM T98311 CGF84D 13500805 IC50 = 6 nM T98311 C4HL9V 13588381 IC50 = 10 nM T98311 C0CY8V 13608313 IC50 = 440000 nM T98311 CW6F9B 13608331 IC50 = 8.1 nM T98311 CY47XT 13652520 IC50 = 10 nM T98311 CW2Y3E 13687301 IC50 = 707.95 nM T98311 CUTA37 13749496 IC50 = 480000 nM T98311 C5WGP2 13749498 IC50 = 19 nM T98311 C69ACG 13749504 IC50 = 10 nM T98311 CUH8T2 14212863 IC50 = 25.12 nM T98311 C81ACD 14212864 Ki = 0.5 nM T98311 CHS29Y 14390729 IC50 = 4 nM T98311 C0N5VL 14540994 IC50 = 200 nM T98311 CZK9D7 14540996 IC50 = 0.5 nM T98311 C8EYH0 14630734 IC50 = 3.236 nM T98311 CO5MX9 14630735 IC50 = 0.4898 nM T98311 CG8S3T 14630739 IC50 = 0.1318 nM T98311 C4IDN0 14630741 IC50 = 338.84 nM T98311 C95DVH 14630745 IC50 = 0.8913 nM T98311 CA59NB 14630749 IC50 = 0.7762 nM T98311 C5GN3K 14630751 IC50 = 0.5248 nM T98311 C3MRF1 14630755 IC50 = 0.5248 nM T98311 C3AV1O 14630757 IC50 = 1.905 nM T98311 C9MA5H 14630761 IC50 = 2.57 nM T98311 CXW6K5 14630765 IC50 = 0.631 nM T98311 CICW62 14630769 IC50 = 0.871 nM T98311 CE1MF9 14630771 IC50 = 15.85 nM T98311 COT04P 14630782 IC50 = 0.2951 nM T98311 CAF28C 14630789 IC50 = 1.072 nM T98311 CYC2U8 14630797 IC50 = 0.2884 nM T98311 CF3TS8 14630801 IC50 = 0.1148 nM T98311 CP73OL 14954082 IC50 = 1995262.31 nM T98311 CLH8D1 15380810 IC50 = 17 nM T98311 CQ20VS 15380813 IC50 = 13 nM T98311 CFX03B 15380816 IC50 = 306 nM T98311 CR40IL 15380817 IC50 = 284 nM T98311 C24BMZ 15380820 IC50 = 4.4 nM T98311 C7R3WN 15380821 IC50 = 28 nM T98311 C93DAN 15615011 IC50 = 2570.4 nM T98311 CQGY31 15838528 IC50 = 33 nM T98311 C9TS8Q 15838530 IC50 = 25 nM T98311 CML3T8 16007169 Ki = 7000 nM T98311 CR0S7G 18542459 IC50 = 1700000 nM T98311 C0SNA2 18601751 IC50 = 10 nM T98311 CSH06N 18608376 IC50 = 7 nM T98311 CFP04Y 18608377 Ki = 11 nM T98311 CGT7B1 20285352 IC50 = 48000 nM T98311 C2YAJ0 20336735 IC50 = 2398.83 nM T98311 C72UNP 20430901 IC50 = 158.49 nM T98311 C1ZUJ8 20430909 IC50 = 63.1 nM T98311 C5YH9C 20430913 IC50 = 125.89 nM T98311 CZ0EC4 20445899 IC50 = 7.943 nM T98311 CZ63YJ 20557515 IC50 = 3.162 nM T98311 CSM6K5 20834249 IC50 = 5.248 nM T98311 CIAR58 21152492 IC50 = 7943.28 nM T98311 C9C3UX 21319418 IC50 = 260000 nM T98311 C7E1XV 21967878 IC50 = 3000 nM T98311 C04LJH 21967881 IC50 = 420 nM T98311 CV8W1T 22799800 IC50 = 64.57 nM T98311 CK6TS0 22805094 IC50 = 229086.77 nM T98311 CSJ07X 22818650 IC50 = 3.7 nM T98311 CF3IS9 22823240 IC50 = 48.98 nM T98311 CU1G0L 22824107 IC50 = 34.67 nM T98311 CFW85M 23322524 IC50 = 4.8 nM T98311 COX68N 23330158 IC50 = 31.62 nM T98311 CBXC05 24424330 IC50 = 0.7 nM T98311 CSWU42 24721360 IC50 = 200 nM T98311 C2MV9X 24882714 IC50 = 1980 nM T98311 CP2LY7 25033280 Ki = 200 nM T98311 C4YKQ1 25033281 Ki = 2700 nM T98311 CR16ZF 25108825 IC50 = 31000 nM T98311 CUC8N5 25141405 IC50 > 100000 nM T98311 CJ0CE4 36688130 IC50 = 6100 nM T98311 C7F3QA 40458146 IC50 = 616595 nM T98311 CT9M6L 40532589 IC50 = 1096478.2 nM T98311 CCH0E2 44266573 IC50 = 3 nM T98311 CXM53J 44266591 IC50 = 7.6 nM T98311 CH7F1P 44266803 IC50 = 1600 nM T98311 CC6SU7 44266804 IC50 = 100000 nM T98311 CY1N3U 44266843 IC50 = 11 nM T98311 CVF0N1 44266856 IC50 = 22000 nM T98311 C6BS5J 44278891 IC50 = 67000 nM T98311 CZ0K4Q 44280449 IC50 = 40.74 nM T98311 CKJ6D4 44288065 IC50 = 13 nM T98311 C1K9TL 44295879 IC50 = 14 nM T98311 C7ZK6W 44295891 IC50 = 36 nM T98311 CSE6U2 44295892 IC50 = 36 nM T98311 CQ07SX 44295893 IC50 = 36 nM T98311 C3G2VM 44295920 IC50 = 183 nM T98311 C6Y1TE 44295939 IC50 = 6.3 nM T98311 C62VIB 44295941 IC50 = 24 nM T98311 CDF39L 44295958 IC50 = 5.4 nM T98311 CFIG72 44295966 IC50 = 14 nM T98311 C6MXZ5 44295979 IC50 = 22 nM T98311 C9F2HK 44296019 IC50 = 18 nM T98311 CD9M3U 44296036 IC50 = 13 nM T98311 C5Z6AR 44296037 IC50 = 31 nM T98311 C0O2CV 44298205 IC50 = 2900 nM T98311 C5D0NQ 44298316 IC50 = 4000 nM T98311 CEU45Z 44298353 IC50 = 4000 nM T98311 CB4PE3 44298355 IC50 = 3600 nM T98311 CJBL20 44298400 IC50 = 4400 nM T98311 CH02UQ 44298401 IC50 = 4000 nM T98311 CL5H7U 44298402 IC50 = 3400 nM T98311 C5G3NH 44298403 IC50 = 800 nM T98311 CUC17Z 44298425 IC50 = 2400 nM T98311 C6WF0X 44298426 IC50 = 3500 nM T98311 CN5A9C 44298428 IC50 = 3500 nM T98311 C14KEU 44298431 IC50 = 2800 nM T98311 CP96RN 44298467 IC50 = 3500 nM T98311 CAQ3R9 44298529 IC50 = 8000 nM T98311 C28WVO 44298544 IC50 = 3800 nM T98311 CB6G8U 44301397 IC50 = 22000 nM T98311 CO53EW 44301408 IC50 = 24000 nM T98311 CGZ1U8 44301409 IC50 > 100000 nM T98311 CC9SL1 44301410 IC50 = 49000 nM T98311 CE9X0Y 44301492 IC50 = 58000 nM T98311 CRB40W 44301493 IC50 = 14000 nM T98311 CJA5G4 44301514 IC50 = 520 nM T98311 CJ75TA 44301544 IC50 = 5.8 nM T98311 C5PY9V 44301552 IC50 = 3.1 nM T98311 CWYK75 44301553 IC50 > 10000 nM T98311 CKX6U5 44301557 IC50 = 58000 nM T98311 C06JQA 44301623 IC50 = 440 nM T98311 CR1M7T 44303110 Ki = 1.3 nM T98311 CW2Y0P 44305060 IC50 = 4900 nM T98311 C73KWG 44305071 IC50 = 50000 nM T98311 CN5YE7 44305121 IC50 = 16 nM T98311 C35AID 44305131 IC50 = 6 nM T98311 CEM4D9 44305132 IC50 = 10 nM T98311 CVS47D 44305140 IC50 = 60 nM T98311 C5D2WT 44305173 IC50 = 20 nM T98311 C45NAZ 44305193 IC50 = 7 nM T98311 CCEN18 44305370 IC50 = 8 nM T98311 C97JBA 44305372 IC50 = 12 nM T98311 CYN2E6 44305391 IC50 = 16 nM T98311 CYU57O 44306009 IC50 = 2398.83 nM T98311 CMC5H9 44314997 Ki = 50000 nM T98311 CNH42V 44316498 IC50 = 30902.95 nM T98311 C31XQM 44316511 IC50 = 645.65 nM T98311 C7BZG0 44316726 IC50 = 1047128.55 nM T98311 CDZ83L 44316727 IC50 = 4570.88 nM T98311 C4R9OS 44316742 IC50 = 389.05 nM T98311 CJC68P 44316752 IC50 = 239883.29 nM T98311 CW7X4R 44316753 IC50 = 3.02 nM T98311 CGS02L 44316769 IC50 = 2.884 nM T98311 CR3U4H 44316777 IC50 = 47863.01 nM T98311 CRS6V0 44316778 IC50 = 8317.64 nM T98311 C0H5KE 44316798 IC50 = 2.884 nM T98311 CO47CU 44316799 IC50 = 100 nM T98311 C9HZU0 44316829 IC50 = 323.59 nM T98311 CD42LH 44316833 IC50 = 77624.71 nM T98311 C5UZ3C 44316834 IC50 = 3467368.5 nM T98311 C90GVY 44316848 IC50 = 2511.89 nM T98311 CF19MI 44316849 IC50 = 12.02 nM T98311 CSJW52 44316850 IC50 = 51.29 nM T98311 CH0R6M 44316851 IC50 = 2.188 nM T98311 C91UJF 44316862 IC50 = 2.188 nM T98311 C9XIC1 44316863 IC50 = 1.096 nM T98311 CSR42L 44316995 IC50 = 218.78 nM T98311 C98RBX 44316996 IC50 = 100 nM T98311 C83GOT 44317006 IC50 = 1819700.86 nM T98311 CET86Y 44317007 IC50 = 758.58 nM T98311 C17PCE 44317014 IC50 = 0.6026 nM T98311 CE0F4B 44317022 IC50 = 15.14 nM T98311 CTPG34 44317023 IC50 = 3.467 nM T98311 CP1ZD0 44317024 IC50 = 0.2512 nM T98311 CREQ84 44317041 IC50 = 38018.94 nM T98311 CP96IH 44317066 IC50 = 2511.89 nM T98311 CLAI57 44317085 IC50 = 25703.96 nM T98311 CFYZ13 44317098 IC50 = 12.02 nM T98311 C97MLC 44317099 IC50 = 2570.4 nM T98311 CV9GO2 44317115 IC50 = 1584.89 nM T98311 CLHB32 44317122 IC50 = 52.48 nM T98311 CP6FN2 44317123 IC50 = 4.786 nM T98311 C90MCR 44317124 IC50 = 0.2291 nM T98311 CM1WH6 44317125 IC50 = 3.02 nM T98311 C63XOZ 44317140 IC50 = 56.23 nM T98311 CUS01W 44317141 IC50 = 436.52 nM T98311 C5Y9TJ 44317145 IC50 = 50.12 nM T98311 C0CQ9A 44317192 IC50 = 4897.79 nM T98311 CQ5F2W 44317193 IC50 = 10232.93 nM T98311 C9LV6D 44317202 IC50 = 64.57 nM T98311 CCK6Q5 44317203 IC50 = 8.913 nM T98311 CE7UV6 44317220 IC50 = 2.57 nM T98311 C05DXW 44317221 IC50 = 63.1 nM T98311 CKDQ56 44317244 IC50 = 2.818 nM T98311 CW5XS4 44317245 IC50 = 645654.23 nM T98311 CL7HU2 44317255 IC50 = 5754.4 nM T98311 CG4MD7 44317265 IC50 = 489778.82 nM T98311 C5VC9Y 44317282 IC50 = 933254.3 nM T98311 CR36KD 44317350 IC50 = 70.79 nM T98311 CYJ4H5 44317359 IC50 = 707.95 nM T98311 CQWT76 44317367 IC50 = 6.457 nM T98311 C43PFU 44321145 IC50 = 12000 nM T98311 COQC17 44321532 IC50 = 1700 nM T98311 C6F5YM 44323100 IC50 = 43 nM T98311 C27WIV 44323101 IC50 = 253 nM T98311 CF2TC5 44323117 IC50 = 42 nM T98311 C2LQX9 44323123 IC50 = 506 nM T98311 CEV4C0 44323191 IC50 = 147 nM T98311 CJW7H8 44323192 IC50 = 18 nM T98311 C6UH2T 44323289 IC50 = 696 nM T98311 CB9PO2 44324428 IC50 > 1000 nM T98311 C3F8DZ 44324530 IC50 = 60 nM T98311 CG6M1Z 44324624 IC50 = 181970.09 nM T98311 CBF46I 44324644 IC50 > 1000 nM T98311 C0Y8EC 44324645 IC50 = 385 nM T98311 CF9M7Y 44324653 IC50 > 1000 nM T98311 CK4R2O 44324830 IC50 = 23 nM T98311 C0O3FJ 44324831 IC50 = 22 nM T98311 C0A8MV 44324877 IC50 = 50 nM T98311 CP6K4X 44325010 IC50 > 1000 nM T98311 C92CXR 44325039 IC50 = 660 nM T98311 CJ6VC5 44325055 IC50 = 100 nM T98311 C9KD1P 44325081 IC50 = 147 nM T98311 C2ZG6V 44325082 IC50 = 414 nM T98311 CE0BW7 44325086 IC50 = 240 nM T98311 C6A1TX 44325087 IC50 = 122 nM T98311 CNHV10 44325092 IC50 = 117 nM T98311 C78HBX 44325093 IC50 = 731 nM T98311 CFNJ58 44325094 IC50 > 1000 nM T98311 CDMZ17 44325095 IC50 = 665 nM T98311 C1V3HD 44325102 IC50 = 65 nM T98311 CNT5D4 44325166 IC50 = 53 nM T98311 C0LH2X 44325169 IC50 = 473 nM T98311 C9ZX5S 44325207 IC50 = 44 nM T98311 CO0S6K 44325221 IC50 > 1000 nM T98311 C24XTA 44325222 IC50 = 138 nM T98311 CX70LB 44325223 IC50 > 1000 nM T98311 CK4XN1 44325232 IC50 = 160 nM T98311 C3J1QZ 44325246 IC50 > 1000 nM T98311 CAI35V 44325247 IC50 = 498 nM T98311 CMZY36 44325303 IC50 > 1000 nM T98311 CSQ37C 44328852 IC50 = 3200 nM T98311 CHA38L 44331702 IC50 = 3.5 nM T98311 CA85MQ 44331737 IC50 = 10000 nM T98311 C0M1RW 44331738 IC50 = 1500 nM T98311 CH8J1T 44336332 Ki = 10 nM T98311 CHD7M2 44337491 IC50 = 5.012 nM T98311 CO6VY1 44337754 IC50 = 3.162 nM T98311 CZ0JK8 44337769 IC50 = 0.7943 nM T98311 C80QCV 44337791 IC50 = 1000000000 nM T98311 CL7K4N 44342229 IC50 > 10000 nM T98311 CC0AG1 44342309 IC50 = 12 nM T98311 CJXP15 44342310 IC50 = 5 nM T98311 C3UHG6 44342481 Ki = 9.8 nM T98311 CEF4J6 44352073 IC50 = 0.6 nM T98311 C6CXD9 44352086 IC50 = 650 nM T98311 C9O7JL 44352389 IC50 = 4200 nM T98311 C4UO8R 44352399 IC50 = 700 nM T98311 C7U0CW 44352420 IC50 = 78000 nM T98311 CXLY79 44352485 IC50 = 16000 nM T98311 C8Q6EW 44358246 IC50 = 2.9 nM T98311 CTE2I6 44358261 IC50 = 8.5 nM T98311 CN0SF8 44358282 IC50 = 5.4 nM T98311 CUY49T 44358403 IC50 = 2600000 nM T98311 CLA34I 44358418 IC50 = 2.9 nM T98311 C2LW8Z 44358438 IC50 = 6 nM T98311 C0KPL6 44358439 IC50 = 9.4 nM T98311 C2EFO5 44364784 IC50 > 10000 nM T98311 CIG7T5 44364906 IC50 = 6000 nM T98311 CF53QE 44364917 IC50 = 470 nM T98311 CM6IJ8 44365196 IC50 = 500 nM T98311 C8D3EI 44365739 Ki = 1.2 nM T98311 C4XOS3 44368279 IC50 = 2400 nM T98311 C89VPA 44368523 IC50 = 90 nM T98311 CA57WU 44368529 IC50 = 260000 nM T98311 CJ4QN7 44368530 Ki = 50000 nM T98311 CBPH20 44368554 IC50 = 0.6 nM T98311 CG75AN 44377126 Ki = 30 nM T98311 CRP20F 44379187 Ki = 1.7 nM T98311 C7EFO1 44383695 IC50 = 6100 nM T98311 C62UTQ 44383743 IC50 = 2800 nM T98311 CTFS09 44384017 IC50 > 10000 nM T98311 CZ9E1G 44384213 IC50 = 4000 nM T98311 CVQ2L3 44384274 IC50 = 4500 nM T98311 CI49UJ 44384300 IC50 = 710 nM T98311 CU87YQ 44384394 IC50 = 300 nM T98311 CRD20Q 44384569 IC50 = 46 nM T98311 C4YK9Q 44384727 IC50 = 10 nM T98311 CVJX47 44384730 IC50 = 15 nM T98311 CJ38IM 44384776 IC50 = 300 nM T98311 C5C9JP 44384800 IC50 = 42 nM T98311 C1GZ3J 44384859 IC50 = 540 nM T98311 CDCY82 44384897 IC50 = 1.4 nM T98311 CQ0CL7 44384992 IC50 = 240 nM T98311 C0W2QL 44384993 IC50 = 5.7 nM T98311 C25WKD 44385190 IC50 = 1300 nM T98311 C2EN3J 44385237 IC50 = 1600 nM T98311 C20YZG 44385438 IC50 = 28 nM T98311 C12UQD 44385469 IC50 = 1.4 nM T98311 CZS79C 44385470 IC50 = 330 nM T98311 CN9YX0 44385527 IC50 = 180 nM T98311 CEI0L8 44385582 IC50 = 1600 nM T98311 C0HDN6 44385628 IC50 = 20 nM T98311 C4YJ6G 44385749 IC50 = 8600 nM T98311 C9XS5C 44385867 IC50 = 25000 nM T98311 C4K1UD 44386281 IC50 = 82 nM T98311 C38FCS 44386286 IC50 = 150 nM T98311 C9XE5J 44386287 IC50 = 4.7 nM T98311 CA3U8H 44386919 IC50 = 656 nM T98311 CF2I3D 44388021 IC50 = 36600 nM T98311 C1FRV0 44400757 IC50 = 14600 nM T98311 CK79BM 44400838 IC50 > 100000 nM T98311 C8J4XB 44401169 IC50 = 31500 nM T98311 CFON28 44404945 IC50 = 0.11 nM T98311 C2PV3I 44404953 IC50 = 5 nM T98311 C6LC0X 44409992 IC50 = 10000 nM T98311 C6T8MR 44415488 Ki = 26300 nM T98311 C06HJB 44446952 Ki = 490 nM T98311 CNK7X5 44446953 Ki = 250 nM T98311 CEB78N 44446954 Ki = 180 nM T98311 CMO78A 44446956 Ki = 570 nM T98311 CV6H2M 44446957 Ki = 410 nM T98311 CF4KE1 44446959 Ki = 1800 nM T98311 CW9C0E 44446960 Ki = 310 nM T98311 CQB5M0 44446963 Ki = 20000 nM T98311 C94POY 44446965 Ki = 1000 nM T98311 CBX2U9 44446967 Ki = 5000 nM T98311 CRZ6B3 44446968 Ki = 1100 nM T98311 CY9O4I 44446969 Ki = 250 nM T98311 C4PQ7D 44446970 Ki = 770 nM T98311 C96KIY 44446972 Ki = 750 nM T98311 CK1EM5 44446974 Ki = 570 nM T98311 C4V6RZ 44446975 Ki = 4000 nM T98311 CBL9E6 44446976 Ki = 950 nM T98311 CVYX54 44446979 Ki = 1800 nM T98311 CAI9Z6 44446980 Ki = 2600 nM T98311 C86KVP 44446984 Ki = 25000 nM T98311 COYX76 44454536 IC50 = 40 nM T98311 CL15BG 44454596 IC50 = 39 nM T98311 CKO40E 44454648 IC50 = 191 nM T98311 C4XKJ6 44454674 IC50 = 23 nM T98311 C9O5YF 44454700 IC50 = 60 nM T98311 C18UOF 44454730 IC50 = 110 nM T98311 CAS59Y 44454780 IC50 = 103 nM T98311 C10OTH 44454833 IC50 = 29 nM T98311 CYK78A 44454905 IC50 = 150 nM T98311 CC2IS3 44454957 Ki = 13000 nM T98311 C1ESI2 44454959 Ki = 620 nM T98311 C8L0MV 44454960 Ki = 700 nM T98311 CBG6T0 44454987 Ki = 200 nM T98311 CN7UW3 44455013 Ki = 9.3 nM T98311 CC5L7S 44455015 Ki = 3400 nM T98311 C6KDT1 44455016 Ki = 8.6 nM T98311 CF4ML7 44455018 Ki = 21 nM T98311 CZI6S1 44455047 Ki = 16 nM T98311 C3UF6E 44455406 Ki = 93 nM T98311 CJG71N 44455407 Ki = 210 nM T98311 C0IR5W 44455428 Ki = 840 nM T98311 C62KSV 44455429 Ki > 10000 nM T98311 CR9WL2 44455430 Ki = 3.2 nM T98311 C6XCJ1 44459080 IC50 = 70000 nM T98311 C31XOD 44459545 IC50 = 110 nM T98311 CR6SJ8 44459614 IC50 = 86 nM T98311 C98LAZ 44459680 IC50 = 14 nM T98311 C1QM5C 44459870 IC50 = 2900 nM T98311 CYTE02 44459897 IC50 = 24 nM T98311 C6XD8J 44459908 IC50 = 220 nM T98311 C15PBV 44461233 IC50 = 290 nM T98311 C25YOU 44461318 IC50 = 3100 nM T98311 CIT5G7 44561891 IC50 > 100000 nM T98311 C90BGR 44561892 IC50 > 100000 nM T98311 C9RGX4 44561893 IC50 > 100000 nM T98311 CU7NP5 44561930 IC50 > 100000 nM T98311 CV21IQ 44561931 IC50 > 100000 nM T98311 CR08WA 44561932 IC50 > 100000 nM T98311 C7H4FK 44581551 IC50 = 100 nM T98311 CM67HS 44581552 IC50 = 250 nM T98311 C2UF1V 44581553 IC50 = 280 nM T98311 CG1VM3 44581554 IC50 = 240 nM T98311 C06ZSJ 44581555 IC50 = 340 nM T98311 C30EFL 44581584 IC50 = 21 nM T98311 CZ4SI2 44581585 IC50 = 210 nM T98311 C4AW6J 44581586 IC50 = 300 nM T98311 CD5EV1 44581587 IC50 = 130 nM T98311 CWI5O1 44581588 IC50 = 280 nM T98311 CL98VN 44581589 IC50 = 4000 nM T98311 CV8CA3 44581623 IC50 = 100 nM T98311 CGOQ13 44581624 IC50 = 260 nM T98311 CH3J8K 44581625 IC50 = 340 nM T98311 C87OUW 44581626 IC50 = 370 nM T98311 CA1TE8 44581627 IC50 = 4600 nM T98311 C9LHM3 44581628 IC50 = 300 nM T98311 CXK2B6 44581658 IC50 = 320 nM T98311 CBZ2Y9 44581659 IC50 = 300 nM T98311 C9DEN6 44581660 IC50 = 300 nM T98311 C8FSX4 44581661 IC50 > 10000 nM T98311 C75IKN 44581662 IC50 = 200 nM T98311 CEF4P5 44581663 IC50 = 340 nM T98311 CV6U4W 44581700 IC50 = 430 nM T98311 CF2YX7 44581701 IC50 = 3600 nM T98311 CFR07N 44581702 IC50 = 1700 nM T98311 CBZ8Q9 44581703 IC50 = 260 nM T98311 C7EK0V 44581746 IC50 > 10000 nM T98311 CL1X5R 44586759 IC50 = 2.4 nM T98311 CEB7D9 44586760 IC50 = 0.18 nM T98311 CMZ46U 44586761 IC50 = 0.029 nM T98311 CXL2R9 44586792 IC50 = 3.2 nM T98311 C9ZCP2 44586816 IC50 = 4.2 nM T98311 C3TN5U 44586817 IC50 = 8.4 nM T98311 CY3OW4 44586818 IC50 = 19 nM T98311 CY4A5N 44586819 IC50 = 15 nM T98311 CH5I4V 44586820 IC50 = 0.9 nM T98311 CMN6G9 44586856 IC50 = 2.3 nM T98311 CRE49N 44586857 IC50 = 4.1 nM T98311 CQAG69 44586858 IC50 = 410 nM T98311 CJA8U3 44586859 IC50 = 280 nM T98311 CQ8T1C 44586860 IC50 = 3.3 nM T98311 CA1YC9 44626604 Ki = 1.4 nM T98311 CK6S5H 44626708 Ki = 3.6 nM T98311 C0EJ1F 44626709 Ki = 0.4 nM T98311 CZR23J 44626710 Ki = 3.8 nM T98311 CQB06H 44626711 Ki = 0.41 nM T98311 C17IGS 44627959 Ki = 13 nM T98311 CM1DL3 44627960 Ki = 5 nM T98311 CNZ8L0 44628063 Ki = 20 nM T98311 CRU86P 44628064 Ki = 25 nM T98311 CS5BG9 44628065 Ki = 12 nM T98311 C65RAJ 45102601 IC50 > 10000 nM T98311 C03HVM 45267758 IC50 = 830 nM T98311 CJ73YP 45267767 IC50 = 160 nM T98311 CG80EY 45269496 IC50 = 280 nM T98311 CT15VE 45270333 IC50 = 400 nM T98311 C48XKY 45272068 IC50 = 300 nM T98311 CX4DS1 45273826 IC50 = 1010 nM T98311 CTOA14 45485236 Ki = 16 nM T98311 CJH50R 49797481 IC50 > 100000 nM T98311 CN12AO 53353383 IC50 = 158 nM T98311 C51GUC 53354365 IC50 = 51 nM T98311 CRJ5P9 53354369 IC50 = 279 nM T98311 C4G2HT 53354470 IC50 = 8.6 nM T98311 C9NE6D 54039314 IC50 = 7.7 nM T98311 CR8M4Y 54082602 IC50 = 17 nM T98311 CCRF59 54268836 IC50 = 330000 nM T98311 CU92WO 54311655 IC50 = 2 nM T98311 C6KH4Z 54395218 IC50 = 700 nM T98311 CBGY97 54468999 IC50 = 44 nM T98311 CO8BM6 54560245 IC50 = 3 nM T98311 C2L5QR 54587395 Ki = 0.16 nM T98311 CGH0S7 54589400 IC50 > 100000 nM T98311 C3S0IT 57393223 IC50 = 580 nM T98311 CC2P9X 57394944 IC50 = 140 nM T98311 CF54YD 57396692 IC50 = 220 nM T98311 CDFA84 57396694 IC50 = 460 nM T98311 C2QE1B 57396695 IC50 = 4800 nM T98311 CA2D6Y 57398463 IC50 = 2000 nM T98311 C3OR9M 71449055 IC50 = 40 nM T98311 C2JE4T 71449056 IC50 = 1400 nM T98311 CUG54A 71454428 IC50 = 4.8 nM T98311 CF6S3Y 71456660 Ki = 3 nM T98311 CY6L9B 71459996 IC50 > 1000 nM T98311 CMF80T 71461712 IC50 = 1100 nM T98311 C4FWY1 71462052 IC50 = 12 nM T98311 C3PU7K 71718514 IC50 = 1.2 nM T98311 C1CKV6 71750764 IC50 = 90000 nM T98311 CA29QZ 72697595 IC50 = 40 nM T98311 CT2MS6 72697596 IC50 = 30 nM T98311 CJXR64 90655798 Ki = 21 nM T98311 CXP0U7 90655799 IC50 = 52 nM T98311 C0XQW8 90655800 IC50 = 220 nM T98311 C54ESG 90668209 IC50 > 31622.78 nM T98311 CX4MK8 90668210 IC50 > 31622.78 nM T98311 CX5MA6 90668211 IC50 > 31622.78 nM T98311 C3YZO5 90668278 IC50 > 31622.78 nM T98311 C8LC4Z 118718824 IC50 = 92 nM T98311 CC80MR 122179189 IC50 = 113000 nM T98311 C2A7DH 122179190 IC50 = 347000 nM T98311 C9QKI3 127020966 IC50 > 100000 nM T98311 CJ98CG 132451821 Ki = 7400 nM T98311 CJZ9I0 145949262 IC50 = 460000 nM T98311 CXE5B0 145949765 IC50 = 2.846 nM T98311 C3P4CF 145951239 IC50 = 7.64 nM T98311 CG1W2X 145951970 IC50 = 9.82 nM T98311 C8WMN6 145952431 IC50 = 11.8 nM T98311 CQ35SP 145953190 IC50 = 10.67 nM T98311 CVUC48 145953329 IC50 = 24.22 nM T98311 CXY8W2 145953611 IC50 = 18.97 nM T98311 C6MTC3 145957046 IC50 = 22.3 nM T98311 C5D9GN 145958042 IC50 = 15.11 nM T98311 CE41NM 145958358 IC50 = 112 nM T98311 CA7YZ0 145959902 IC50 = 4.11 nM T98311 CE72UY 145963315 IC50 = 8.841 nM T98311 C7JFL1 145984090 IC50 = 43 nM T98311 CFXM92 145994098 IC50 = 2100 nM T98311 CU42CE 155567829 IC50 > 100000 nM T98311 D00KEP 6049 IC50 = 14000 nM T98311 D02BTV 9816867 IC50 > 100000 nM T98311 D02FMN 9827219 Ki = 7 nM T98311 D02NQB 10430040 IC50 > 100000 nM T98311 D03QJA 11718722 IC50 = 193 nM T98311 D03SPJ 73568 IC50 = 3700000 nM T98311 D03UIF 9906720 IC50 = 520 nM T98311 D07APP 131255 IC50 = 13400 nM T98311 D08ELY 9838786 IC50 = 81000 nM T98311 D0A1CM 5281855 IC50 = 5000000 nM T98311 D0B3UN 44580458 Ki > 100000 nM T98311 D0C6QS 3001497 IC50 = 400000 nM T98311 D0G3YZ 11391583 IC50 > 250000 nM T98311 D0K0OY 44346192 Ki = 100 nM T98311 D0N4RO 44377139 Ki = 520 nM T98311 D0N6CD 10565532 IC50 > 100000 nM T98311 D0N8YA 159596 IC50 > 100000 nM T98311 D0PB5Q 3132 IC50 = 316.23 nM T98311 D0Y3TZ 370 IC50 = 7700000 nM T98311 D0Y5IQ 44255320 IC50 = 10000 nM T54156 D00HNB 25419 IC50 = 320000 nM T54156 D00MDP 466151 IC50 = 0.2 nM T54156 D04AIT 5280445 IC50 = 5620 nM T54156 D0K8KX 5280343 IC50 = 1610 nM T54156 D0Q8CS 60937 IC50 > 100000 nM T54156 D0V4GY 9552079 IC50 = 7630 nM T54156 D0VM2L 68740 IC50 = 52000 nM T54156 D04LTF 9868980 IC50 = 0.6 ug.mL-1 T54156 D05VZE 119031 Ki < 1 nM T54156 D0F2JS 15547703 IC50 = 1500 nM T54156 D0MW3H 9824350 IC50 = 2.4 nM T54156 D0N4IV 10718956 IC50 = 9.6 nM T54156 D09EFW 46861776 IC50 = 3.33 nM T54156 D00UCC 9827497 IC50 = 0.5 nM T54156 D01DVX 9847838 IC50 = 389 nM T54156 D03BOZ 3342298 IC50 = 0.11 nM T54156 D0E5GY 9904965 Ki = 2 nM T54156 D0P8YC 5362422 IC50 = 0.6 nM T54156 D0Q1CD 6918336 Ki = 301 nM T54156 D0T9HG 132519 IC50 = 0.05 nM T54156 D0Y1XT 128564 Ki < 1 nM T54156 CNA81R 1836 Ki = 52 nM T54156 CY78XM 4218 IC50 = 1.8 nM T54156 CFY8Q2 4230 IC50 = 1.9 nM T54156 CL2W6Q 38422 IC50 > 20000 nM T54156 CPW9B5 65752 IC50 = 7.95 ug.mL-1 T54156 CYEU83 69033 Ki = 78000 nM T54156 C0PY5N 77754 Ki > 100 nM T54156 CR37WJ 115121 IC50 = 5.8 ug.mL-1 T54156 CP4O2C 121255 Ki = 66000 nM T54156 CDJS43 154136 IC50 = 3.9 nM T54156 C50IPY 154137 IC50 = 4.7 nM T54156 CCY6L8 169853 IC50 = 53200 nM T54156 C7ROG5 177347 IC50 = 3110 nM T54156 CJ62BZ 193987 IC50 = 59 nM T54156 CP7Q8T 240910 Ki = 24000 nM T54156 CX3DK6 283995 Ki = 10000 nM T54156 COFX01 352863 Ki = 76000 nM T54156 CK9M3P 445018 IC50 = 6.8 nM T54156 C4D7TS 448002 IC50 = 4.8 nM T54156 CC54LQ 450256 IC50 > 100000 nM T54156 C45JSH 639942 IC50 = 6.19 nM T54156 CCKZ79 668744 IC50 = 43000 nM T54156 CP91NX 677915 IC50 = 1812.91 nM T54156 CDE9V2 689424 IC50 = 1896.92 nM T54156 C5O0TJ 690158 IC50 = 7.98 nM T54156 C7TPR6 690965 IC50 = 6.21 nM T54156 C9FL2X 721434 IC50 = 1796.72 nM T54156 CTO15S 727131 IC50 = 10.26 nM T54156 CTV50K 727184 IC50 = 1910.47 nM T54156 C2CL6X 732134 IC50 = 7.29 nM T54156 CPKI76 765318 IC50 = 13.87 nM T54156 CXME85 766168 IC50 = 12.59 nM T54156 CWQG91 770865 IC50 = 3400 nM T54156 CQB03J 780790 IC50 = 7.38 nM T54156 C7EHR1 787183 IC50 = 6.38 nM T54156 C5MF2E 795596 IC50 = 1976.83 nM T54156 C1K0NF 795855 IC50 = 8.19 nM T54156 CW56XG 875024 IC50 = 10.58 nM T54156 C17IXT 910211 IC50 = 8.13 nM T54156 C8A5CX 1800786 IC50 > 10000 nM T54156 C36DGS 2211098 IC50 = 180 nM T54156 CN6E3U 2366268 IC50 = 2200 nM T54156 CN62WX 2800809 IC50 = 6000 nM T54156 CY3TD6 3348132 Ki = 10 nM T54156 CME24U 3649035 IC50 > 101000 nM T54156 CBN96T 4358655 IC50 > 100000 nM T54156 CC5O4E 4369384 IC50 = 2000 nM T54156 CZBY34 5220706 Ki = 69000 nM T54156 C20HRJ 5273475 IC50 = 7.18 nM T54156 CZS0G5 5276565 IC50 > 100000 nM T54156 C3JN0F 5277465 IC50 > 100000 nM T54156 CRJK67 5277481 IC50 > 100000 nM T54156 CYF7S5 5277490 IC50 > 100000 nM T54156 CJ3QI1 5288814 IC50 = 1390 nM T54156 CO58XD 5311161 IC50 > 100000 nM T54156 CVLS16 5319161 IC50 = 11610 nM T54156 CDI23X 5941957 IC50 > 100000 nM T54156 C4J3PG 6250177 IC50 = 60100 nM T54156 C0M3LR 6323382 IC50 = 71 nM T54156 CND9M2 6449880 IC50 = 13400 nM T54156 CJG2B7 6476333 IC50 = 14280 nM T54156 CL5DH0 6479915 IC50 = 610 nM T54156 CQEF36 6539670 IC50 = 0.54 nM T54156 CN5L2B 6852147 IC50 = 8 nM T54156 CPFV65 6916013 Ki = 125.89 nM T54156 CG2A7X 7028541 IC50 = 105900 nM T54156 C7Y1BX 9543420 IC50 = 20.6 nM T54156 CIJ25V 9794947 IC50 > 100000 nM T54156 CLK61C 9797144 Ki = 162 nM T54156 CA0ZH1 9798114 IC50 = 777 nM T54156 C7NP9Z 9798247 IC50 = 62 nM T54156 C78EKW 9798637 IC50 = 14 nM T54156 C76RCQ 9801569 IC50 = 591 nM T54156 CM9GH8 9802180 IC50 = 1.4 nM T54156 CJY12B 9802219 Ki > 2000 nM T54156 C4CN0H 9802436 Ki = 0.097 nM T54156 CIXD67 9802768 IC50 = 1.5 nM T54156 C83FVW 9803207 IC50 = 1 nM T54156 C3QS5H 9803407 IC50 = 148 nM T54156 C4QCG9 9803771 IC50 = 14 nM T54156 C49HNU 9805016 IC50 = 3 nM T54156 CP65QD 9805079 Ki > 2000 nM T54156 CXSU10 9805304 IC50 = 477 nM T54156 CO4D0U 9805473 IC50 = 1 nM T54156 C1HP7E 9805710 IC50 = 3.6 nM T54156 CT8X1F 9806970 IC50 = 857 nM T54156 C76CKA 9807105 Ki > 2000 nM T54156 CTK6J8 9808181 IC50 = 30400 nM T54156 C67XKV 9808391 IC50 = 2 nM T54156 CS07BM 9808594 IC50 = 3 nM T54156 C9RQM7 9808674 IC50 = 0.1 nM T54156 CTO36D 9817594 IC50 > 100000 nM T54156 CC9VY4 9819420 IC50 = 364 nM T54156 C1VT4J 9819974 IC50 = 170 nM T54156 CQG86S 9820708 IC50 = 10 nM T54156 C5OE1B 9821883 Ki = 27 nM T54156 CJC20A 9822095 IC50 = 30 nM T54156 C6KJ9W 9822461 IC50 = 21 nM T54156 C6IX7G 9822926 IC50 = 0.3 nM T54156 C1MPW9 9823182 IC50 = 17 nM T54156 CTF8V4 9823391 Ki > 2000 nM T54156 CUZ25T 9825237 IC50 = 33 nM T54156 C3AEF4 9825692 IC50 = 19 nM T54156 CDJB86 9825720 IC50 = 0.6 nM T54156 CXL65P 9825920 Ki > 2100 nM T54156 C65ZHY 9826199 IC50 = 0.32 nM T54156 CVSJ72 9826275 IC50 = 3 nM T54156 C7W3TG 9826481 IC50 = 800 nM T54156 CPW60S 9827023 IC50 = 95.5 nM T54156 CXTY18 9827218 IC50 = 70 nM T54156 C1A7NJ 9827355 Ki = 1.9 nM T54156 C3SZ8Y 9827469 Ki > 2000 nM T54156 C2TU0C 9827807 IC50 = 4 nM T54156 CL59JS 9827846 IC50 = 13 nM T54156 C7I2FO 9828039 Ki = 291 nM T54156 C1GR4N 9828276 IC50 > 25000 nM T54156 CC1NG5 9829581 IC50 = 8 nM T54156 C7SRM4 9837496 IC50 > 100000 nM T54156 C8WH1Q 9840355 IC50 = 11 nM T54156 CU7FM2 9840390 IC50 = 484 nM T54156 CEAZ87 9840395 IC50 = 111 nM T54156 CKF84D 9840581 IC50 = 8 nM T54156 C9PW7L 9841168 Ki = 446.7 nM T54156 CQ5L0D 9842167 IC50 = 2500 nM T54156 CH63ZI 9842332 IC50 = 21 nM T54156 CC1TB5 9842343 IC50 = 649 nM T54156 C32JRZ 9843079 IC50 = 50 nM T54156 CK76RW 9845271 IC50 = 138 nM T54156 CEB90C 9846418 IC50 = 4 nM T54156 C8T0BQ 9846437 IC50 = 30.9 nM T54156 CWY1J9 9846501 Ki > 2000 nM T54156 C4D2MY 9846507 IC50 = 34 nM T54156 C0KP9H 9847092 IC50 = 4 nM T54156 CE9AL3 9847113 IC50 = 0.2 nM T54156 CA1IP0 9847191 Ki > 2000 nM T54156 C6SV1X 9847843 IC50 = 9 nM T54156 CG14CO 9848625 IC50 = 232 nM T54156 C92EJW 9849379 IC50 = 20 nM T54156 CX3EW2 9849576 IC50 = 385 nM T54156 CHVL24 9849957 IC50 = 3 nM T54156 C4IEK0 9850035 IC50 = 0.25 nM T54156 C9P1BH 9851086 IC50 = 2 nM T54156 C7UP3K 9857957 IC50 = 370 nM T54156 CC70WV 9858468 IC50 = 1262 nM T54156 CR37HQ 9861014 IC50 = 1511 nM T54156 CTY26D 9861878 IC50 = 1000 nM T54156 C5TUJ7 9862317 IC50 = 82 nM T54156 C8CEJ4 9862349 IC50 = 8 nM T54156 C8GE7U 9862764 IC50 = 118 nM T54156 CS5JT6 9864502 IC50 = 56 nM T54156 CU51IV 9865936 IC50 = 10 nM T54156 CI8Z0R 9866250 IC50 = 12 nM T54156 CR10NL 9866770 Ki > 2000 nM T54156 CP4Y7O 9867411 IC50 = 51 nM T54156 CX57RB 9868249 Ki > 2000 nM T54156 C2L9SU 9868329 IC50 = 2 nM T54156 CJS23I 9868333 Ki > 2128 nM T54156 C5O0GC 9868490 IC50 = 221 nM T54156 CRI23M 9868515 IC50 = 15 nM T54156 C4K2GH 9868577 IC50 = 5 nM T54156 CJ8DP1 9868672 IC50 > 6000 nM T54156 C4ZR7O 9868713 IC50 = 228 nM T54156 C5IJH2 9869068 IC50 = 13 nM T54156 CT76IN 9869441 IC50 = 6 nM T54156 CLQ29X 9869597 IC50 = 406 nM T54156 CA6G0W 9869598 IC50 = 5 nM T54156 CG17NZ 9869811 IC50 = 120 nM T54156 CZO6K4 9869819 IC50 = 0.6 nM T54156 C5ELS6 9869902 IC50 = 10 nM T54156 C38BVX 9870100 IC50 = 32 nM T54156 CZO2I0 9870133 IC50 = 15 nM T54156 CA48SX 9870269 IC50 = 3 nM T54156 C25-SEP 9870933 IC50 = 389 nM T54156 C5QFG1 9871290 IC50 = 3 nM T54156 CD1XQ2 9871305 IC50 = 1.1 nM T54156 CHU9I8 9871883 IC50 = 0.15 nM T54156 C5NM6P 9872886 IC50 = 5 nM T54156 CU9L3X 9879183 IC50 > 10000 nM T54156 C0TCJ2 9880675 Ki > 2128 nM T54156 C0NA6S 9880842 IC50 = 107 nM T54156 CW8IC4 9882151 IC50 > 100000 nM T54156 C0ZT7A 9883002 Ki = 400 nM T54156 C2OHV3 9885051 IC50 = 374 nM T54156 C75DAZ 9885136 IC50 = 0.8 nM T54156 CKFD90 9885716 IC50 = 452 nM T54156 CZBK85 9886177 IC50 = 18 nM T54156 C2M4EC 9887473 Ki > 2128 nM T54156 C4PB5Z 9887544 Ki = 1.8 nM T54156 CFG4Q2 9887831 IC50 = 71 nM T54156 C3ZG6O 9887870 IC50 = 7900 nM T54156 CC87LP 9888280 IC50 = 17 nM T54156 C8AJB7 9888429 Ki > 2000 nM T54156 CD76WB 9888485 IC50 = 16 nM T54156 CJS0E5 9888649 IC50 = 23 nM T54156 CHB65O 9889042 IC50 = 104 nM T54156 CB2YG7 9889128 IC50 = 12 nM T54156 CD1U5P 9889190 IC50 = 553 nM T54156 CZD2E3 9889870 IC50 = 44 nM T54156 C26SZX 9890226 IC50 = 0.6 nM T54156 CD79UJ 9890632 IC50 = 61000 nM T54156 CNX78A 9890733 IC50 = 1 nM T54156 CMD0S2 9891009 IC50 = 15 nM T54156 C20LGF 9891255 IC50 = 21 nM T54156 C9YD2O 9891259 IC50 = 11 nM T54156 CU65HY 9891358 IC50 = 0.5 nM T54156 C3QSE6 9891814 IC50 = 2.9 nM T54156 CPT4C6 9892042 IC50 = 236 nM T54156 C1KV7J 9892518 IC50 = 18 nM T54156 CH69LT 9892815 IC50 = 0.18 nM T54156 CZU7Y4 9892876 IC50 = 13 nM T54156 CK1F3O 9892889 Ki > 2000 nM T54156 C2G5AQ 9894201 IC50 = 1205 nM T54156 CSIB97 9896504 IC50 > 100000 nM T54156 C6Q4JF 9903007 IC50 = 38 nM T54156 C97GSC 9903557 Ki > 2128 nM T54156 CD78ZQ 9907286 IC50 = 13 nM T54156 CYHN04 9908006 IC50 = 39 nM T54156 CMSC52 9908418 Ki > 800 nM T54156 CKWF30 9908681 IC50 = 88 nM T54156 C4E6LR 9910544 IC50 = 244 nM T54156 C6NUE9 9910550 IC50 = 1 nM T54156 CT50EC 9912183 Ki > 2000 nM T54156 C2GMQ0 9912235 IC50 = 251 nM T54156 C62VZI 9912382 IC50 = 2.5 nM T54156 C8VJ9Z 9913053 IC50 = 3 nM T54156 CI5A3G 9913301 IC50 = 11 nM T54156 CX1Q5C 9913489 IC50 = 5 nM T54156 CSZV76 9913881 IC50 = 25 nM T54156 C7ZY1L 9914029 IC50 = 26 nM T54156 CU9B3E 9914147 IC50 = 24 nM T54156 CM39FU 9915194 IC50 = 2827 nM T54156 CM7UO8 9924798 IC50 = 9 nM T54156 CBPD13 9926779 IC50 = 18 nM T54156 CSA12Z 9927353 IC50 = 53 nM T54156 C4YGT6 9928325 IC50 = 3.9 nM T54156 C26ZPC 9929976 IC50 = 43 nM T54156 C7EIX4 9930068 Ki = 2.6 nM T54156 CLJ61Q 9931505 IC50 = 28 nM T54156 CJI5A7 9932167 IC50 = 2 nM T54156 C03GVA 9932290 Ki = 80 nM T54156 C1I2FW 9932632 Ki > 2000 nM T54156 CT2KM9 9933083 IC50 = 100 nM T54156 CDXR37 9933197 IC50 = 1.2 nM T54156 C2EUL8 9933259 IC50 = 95 nM T54156 C8E3LV 9933622 Ki = 4000 nM T54156 C5E7PR 9933720 Ki = 3.3 nM T54156 CF26MY 9934052 Ki > 2000 nM T54156 CA5V8M 9934053 Ki = 1299 nM T54156 C57WSD 9934240 IC50 = 16 nM T54156 CGJZ78 9934997 IC50 = 33 nM T54156 C65ION 9935032 IC50 = 2.3 nM T54156 C1HRU9 9936228 IC50 = 2.5 nM T54156 CDRC76 9936405 IC50 = 187 nM T54156 CH9G5D 9936469 IC50 = 35.8 nM T54156 C68MQN 9936625 Ki > 2000 nM T54156 C7GJF8 9936712 IC50 = 2 nM T54156 CG38KL 9936728 Ki = 1.2 nM T54156 C12ZGS 9945200 IC50 = 1380.38 nM T54156 C0MLZ6 9945553 IC50 = 3000 nM T54156 C6TH4I 9947270 IC50 > 10000 nM T54156 CSN61C 9948296 Ki > 2128 nM T54156 C16HTN 9948666 IC50 = 309 nM T54156 C52IUJ 9949603 IC50 = 3000 nM T54156 CF1DO9 9950475 Ki > 2000 nM T54156 CQY54S 9952396 IC50 = 5.1 nM T54156 C9OY4Z 9953817 IC50 = 45 nM T54156 C16GIN 9953861 Ki > 2000 nM T54156 CR6EX3 9953909 Ki = 1964 nM T54156 C6GA8D 9954513 IC50 = 13 nM T54156 CH9YL3 9954604 IC50 = 26 nM T54156 C37VXK 9954605 IC50 = 9 nM T54156 C9X0YR 9954867 Ki = 4468 nM T54156 C32HAZ 9954953 Ki = 1.2 nM T54156 CK9HX0 9955125 IC50 = 1.5 nM T54156 CMV37W 9955127 IC50 = 108 nM T54156 CWE6N8 9955640 IC50 = 8 nM T54156 C05HGV 9955795 IC50 = 2.8 nM T54156 C3ZLA1 9956465 IC50 = 164 nM T54156 C3Q2UJ 9956686 IC50 = 0.25 nM T54156 CS73TB 9956692 Ki > 2128 nM T54156 CI5TW9 9956699 IC50 = 2420 nM T54156 C56GFP 9956833 IC50 = 13 nM T54156 CQ80MP 9957107 IC50 = 13 nM T54156 CC4WG3 9957228 Ki > 300000 nM T54156 C5I0VJ 9957500 IC50 = 387 nM T54156 CN76XI 9957653 IC50 = 1 nM T54156 CPJR82 9957875 IC50 = 6 nM T54156 CWE4D3 9958604 IC50 = 6 nM T54156 CVG0O2 9959014 IC50 = 1 nM T54156 CNHT34 9959421 IC50 = 0.7 nM T54156 CV40RB 9960075 Ki > 2128 nM T54156 C9DRB7 9966028 IC50 = 753 nM T54156 CYK75X 9967932 IC50 > 10000 nM T54156 C0HL2X 9976697 IC50 = 1.9 nM T54156 CA0XP7 9977927 Ki = 100 nM T54156 CUA65C 9982414 IC50 = 5.3 nM T54156 CO09PN 9983251 IC50 = 0.9 nM T54156 CJGR30 9983604 IC50 = 5.4 nM T54156 C8IL6Q 9986000 IC50 = 4.5 nM T54156 CO0TX7 9993891 Ki = 9000 nM T54156 C3KX1B 9998685 Ki = 10 nM T54156 C8W5UK 9999879 IC50 = 414 nM T54156 C6TO0A 10001582 Ki = 1.2 nM T54156 CP5N4E 10005114 Ki = 309 nM T54156 C6U3CK 10006134 IC50 = 0.5 nM T54156 CR7T3J 10009978 Ki = 1787 nM T54156 C71YGT 10025307 Ki = 1.2 nM T54156 C6O0MN 10026682 Ki = 9900 nM T54156 C6DGR7 10027203 Ki = 1.698 nM T54156 C4VJX9 10027747 IC50 = 36000 nM T54156 CVG03H 10031524 IC50 = 7.4 nM T54156 C7J9ZF 10039403 IC50 = 655 nM T54156 C1X0SA 10041385 Ki = 104 nM T54156 CPZ4L1 10041481 IC50 = 6 nM T54156 CNA3G4 10042214 IC50 = 119 nM T54156 CO39PK 10042482 Ki = 95.5 nM T54156 CW2MK1 10043732 Ki = 100 nM T54156 C7O8HD 10044261 IC50 = 2.8 nM T54156 CY1J5S 10045091 IC50 = 79 nM T54156 C7CT4E 10045150 IC50 = 1.3 nM T54156 CHF92V 10047100 Ki = 0.72 nM T54156 CCF5Z4 10047585 IC50 = 0.3 nM T54156 C1N9UX 10050222 IC50 = 304 nM T54156 C1G0HE 10051959 IC50 = 30 nM T54156 CZ6R1T 10052198 Ki = 2.7 nM T54156 CSHD67 10054852 IC50 = 0.2 nM T54156 CSW7B3 10067146 Ki = 8 nM T54156 CSG9A5 10073761 Ki = 3.8 nM T54156 CV0I9M 10074738 IC50 = 32 nM T54156 CPS4R9 10076090 IC50 = 1 nM T54156 CJ2H0T 10077849 IC50 = 13 nM T54156 CU7DJ1 10081163 Ki = 60000 nM T54156 CUT28D 10088847 Ki = 165 nM T54156 CLJT42 10091046 Ki = 51.88 nM T54156 CPKC43 10093147 IC50 = 7 nM T54156 C2XV5J 10098250 IC50 = 7.3 nM T54156 C3V2HW 10099112 IC50 = 2300 nM T54156 CMLA47 10099961 IC50 = 4.8 nM T54156 CXV2Y3 10109170 Ki = 702 nM T54156 C0G7IY 10114318 Ki = 170 nM T54156 C9T2AW 10116042 IC50 = 9 nM T54156 C78JHL 10116107 Ki = 240 nM T54156 C4P1LB 10116618 IC50 = 0.3 nM T54156 CU0D4S 10117481 Ki > 2128 nM T54156 CP5L0W 10117663 Ki > 2100 nM T54156 C7OPQ8 10118047 IC50 = 1100 nM T54156 CU3ZM2 10118633 IC50 > 1000 nM T54156 C2F8KW 10119294 IC50 = 2 nM T54156 CPA4R9 10119730 IC50 = 11 nM T54156 C7A8MI 10120093 IC50 = 0.6 nM T54156 C0Q9DW 10120586 IC50 = 6 nM T54156 CT4V0P 10120622 IC50 = 0.86 nM T54156 C0KHW5 10120930 IC50 = 1162 nM T54156 CY2N3D 10127629 Ki > 2130 nM T54156 C1N4MJ 10127670 Ki > 2130 nM T54156 CIL09Z 10127889 Ki > 2130 nM T54156 C07KFI 10128313 Ki > 2130 nM T54156 CB3I6K 10128659 Ki > 2130 nM T54156 C6ZK3A 10128916 Ki > 2130 nM T54156 CS54CQ 10133565 IC50 > 10000 nM T54156 C9EWX5 10135125 IC50 = 63 nM T54156 CDR73P 10135184 Ki > 2128 nM T54156 C7KR3Y 10136680 Ki = 210 nM T54156 CNU93J 10136924 Ki = 160 nM T54156 C1CDF2 10136925 Ki = 50 nM T54156 CJ9EX4 10138303 Ki = 800 nM T54156 C6UXD7 10138936 IC50 = 79 nM T54156 CFXC89 10139040 Ki > 2128 nM T54156 CGC6S5 10139402 Ki > 2128 nM T54156 CP8QV4 10140363 Ki = 1246 nM T54156 CU6Y9T 10140438 Ki > 2128 nM T54156 CE75BY 10140776 Ki > 2100 nM T54156 CIH36M 10141214 IC50 = 930 nM T54156 C5DA1U 10141270 IC50 = 2 nM T54156 C5H1ZM 10141426 IC50 = 2 nM T54156 C6MSI0 10141443 IC50 > 100000 nM T54156 CLXF15 10141613 Ki > 2100 nM T54156 C7VF1K 10141614 Ki > 2100 nM T54156 CWB5O4 10142326 Ki > 2100 nM T54156 CL7P6G 10143019 IC50 = 7.2 nM T54156 CPXB21 10143028 Ki > 2128 nM T54156 C23WZR 10143587 Ki > 2100 nM T54156 CAM6U7 10143672 IC50 = 8 nM T54156 C82SMW 10144091 IC50 = 4 nM T54156 CUG62E 10155007 IC50 > 40000 nM T54156 CLQ89T 10155008 IC50 = 7000 nM T54156 CZW98O 10156375 Ki = 46.7 nM T54156 CPY87U 10158366 IC50 > 10000 nM T54156 CP87UW 10158843 IC50 = 900 nM T54156 CYO8D2 10159633 Ki > 2128 nM T54156 CQ4SJ5 10160197 Ki > 2128 nM T54156 CQ41YI 10161391 Ki > 2128 nM T54156 CCU9S1 10162155 IC50 = 2 nM T54156 C7SXD4 10162245 Ki > 2100 nM T54156 CO6PS3 10162900 Ki = 40 nM T54156 CR5H6E 10163627 Ki > 2128 nM T54156 CI9VJ5 10163857 Ki > 2128 nM T54156 CR17PV 10164205 Ki > 2128 nM T54156 CZO5V4 10164317 IC50 < 0.4 nM T54156 CCM0Y8 10165180 Ki > 2100 nM T54156 CE10MK 10165419 IC50 = 11 nM T54156 CP02FJ 10165420 IC50 = 11 nM T54156 C0K7HT 10165868 IC50 = 2 nM T54156 C5ZO9J 10166232 IC50 = 0.53 nM T54156 CNTC03 10172417 Ki = 4.8 nM T54156 C6IW4O 10173876 Ki > 2130 nM T54156 C4QY3V 10175210 Ki = 2040 nM T54156 C5JM1A 10179045 IC50 = 10000 nM T54156 CCX3T6 10183064 Ki > 15000 nM T54156 CS6X2R 10183408 IC50 = 2 nM T54156 C6OE9H 10183692 IC50 > 10000 nM T54156 CDM94B 10183693 Ki > 2100 nM T54156 CHB2D3 10184071 Ki > 2128 nM T54156 CH04IS 10184457 IC50 = 2 nM T54156 C3E9NF 10184537 Ki > 2100 nM T54156 CTDP62 10184579 Ki > 2100 nM T54156 CXQ8N0 10185100 Ki > 2128 nM T54156 C2OM9G 10186288 IC50 = 8 nM T54156 CK0P3F 10186536 Ki > 2128 nM T54156 CV7YI1 10186544 Ki > 2100 nM T54156 CA9FG4 10187181 IC50 = 3 nM T54156 C51RPY 10195069 Ki > 2130 nM T54156 CY36NO 10196425 Ki > 2130 nM T54156 CVRZ27 10198038 IC50 > 100000 nM T54156 C0U9KC 10199401 IC50 = 83 nM T54156 C5CUM9 10202769 Ki > 2128 nM T54156 CX8BS3 10203685 Ki > 2128 nM T54156 CE1LI3 10204303 Ki = 40 nM T54156 C32RAQ 10204620 Ki > 2100 nM T54156 CQFP69 10206106 Ki = 160 nM T54156 CS1CA5 10207780 Ki = 2100 nM T54156 C4K1MJ 10208262 Ki > 2128 nM T54156 CYE02Q 10209301 IC50 = 2 nM T54156 CV4DG9 10209314 IC50 = 2 nM T54156 CD76KE 10209382 Ki > 2128 nM T54156 C1C7AH 10223757 Ki > 2128 nM T54156 CYG10Z 10223774 Ki > 2128 nM T54156 CV5X8A 10224181 IC50 > 30000 nM T54156 CGKU70 10224396 Ki = 80 nM T54156 CLH71C 10225319 Ki > 2128 nM T54156 C2X1KF 10226116 Ki > 2100 nM T54156 CJ46HR 10227522 IC50 = 4 nM T54156 CUE63Q 10227853 Ki > 2100 nM T54156 C19DFP 10227854 Ki > 2100 nM T54156 CM7B5T 10228228 Ki > 2128 nM T54156 CSDG58 10228529 IC50 = 643 nM T54156 C7T0WH 10229644 IC50 = 50.8 nM T54156 CD2HP3 10230012 Ki > 2100 nM T54156 CLJ3Y9 10230286 IC50 = 4 nM T54156 CCRM18 10231253 IC50 = 0.2 nM T54156 CCTY95 10237492 Ki > 2130 nM T54156 CQH2U3 10238391 IC50 = 700 nM T54156 CCQ9V5 10239716 Ki > 2130 nM T54156 CL67DT 10252311 Ki < 2.1 nM T54156 CQJ0R3 10252900 Ki = 0.63 nM T54156 C2V4MP 10253549 IC50 = 6 nM T54156 CJ3Q8W 10256080 IC50 = 15 nM T54156 C4WV7B 10257654 IC50 = 27 nM T54156 C6EI1N 10262798 Ki = 6000 nM T54156 CJKD83 10268288 IC50 > 10000 nM T54156 C0CE3N 10269452 IC50 = 12000 nM T54156 C0QS9V 10269453 IC50 = 113 nM T54156 CMNA19 10270268 IC50 > 10000 nM T54156 C2MES9 10271604 Ki > 100000 nM T54156 C0K2ES 10273642 Ki > 2128 nM T54156 CJZP24 10273657 Ki > 2128 nM T54156 CK18DB 10273985 Ki > 2128 nM T54156 CGP97S 10274748 Ki = 60 nM T54156 C13NKU 10275545 Ki > 2128 nM T54156 C1NGV9 10276473 Ki > 2128 nM T54156 CES6A5 10276821 Ki = 1511 nM T54156 C1W7SN 10277073 Ki > 2128 nM T54156 CO18TA 10277120 Ki > 2128 nM T54156 C0GU6B 10277568 IC50 = 6 nM T54156 CY6K1G 10277706 Ki > 2100 nM T54156 C9OAE1 10277812 IC50 = 2 nM T54156 C2XU3O 10278147 IC50 = 1.1 nM T54156 C2UAM8 10278729 IC50 = 1 nM T54156 C6KR5M 10278934 IC50 = 6 nM T54156 C3IG0K 10280852 IC50 = 0.2 nM T54156 C80WUO 10282084 IC50 = 0.79 nM T54156 C7TWG0 10289551 Ki > 2130 nM T54156 CJ63ER 10289607 Ki > 2130 nM T54156 CP0I5Y 10291146 IC50 > 10000 nM T54156 CLP72J 10293348 IC50 > 10000 nM T54156 CB82ZF 10294766 IC50 = 120 nM T54156 C89YGA 10295733 Ki > 2128 nM T54156 CDU36Y 10296475 Ki = 320 nM T54156 CTL3Y8 10296608 Ki > 2128 nM T54156 C48IRP 10296785 Ki = 80 nM T54156 CN14MI 10298369 Ki > 2128 nM T54156 CU5E9Z 10299198 Ki = 1447 nM T54156 C25EKM 10299665 Ki > 2100 nM T54156 CQ5BE8 10299709 IC50 = 0.91 nM T54156 C1BR6A 10300063 Ki > 2128 nM T54156 C80VEU 10300077 Ki > 2128 nM T54156 C8U3KW 10301524 IC50 = 1.7 nM T54156 CFAU84 10301584 Ki > 2128 nM T54156 CP5AU1 10302088 Ki > 2128 nM T54156 C63BRA 10303333 IC50 = 0.98 nM T54156 C4R9ZK 10311997 Ki = 85 nM T54156 CE6MB0 10312141 Ki = 138 nM T54156 CP1GW0 10318094 Ki = 0.54 nM T54156 C2U6MY 10318916 Ki = 21 nM T54156 CF4KT9 10320002 Ki > 2128 nM T54156 CJ6XM1 10321516 IC50 = 1 nM T54156 CVKT01 10322744 IC50 = 50 nM T54156 CY08WJ 10322755 Ki > 3000 nM T54156 C50KSE 10323483 IC50 = 9 nM T54156 C9DR2I 10323789 IC50 = 36 nM T54156 CSFZ76 10325592 Ki > 2128 nM T54156 CSG12E 10325620 IC50 = 5 nM T54156 CF5UN8 10326272 IC50 = 15 nM T54156 C5F0RK 10326931 IC50 = 28 nM T54156 CG6NT9 10338869 IC50 = 90 nM T54156 C7UZA4 10340758 IC50 = 3.3 nM T54156 CFO74N 10343375 Ki = 210 nM T54156 CJIW74 10343996 Ki = 0.31 nM T54156 CW1VL2 10345348 IC50 = 101 nM T54156 CPJ1G8 10345717 IC50 = 69 nM T54156 CX8H3Z 10346437 IC50 = 35 nM T54156 C9FU5G 10362663 IC50 = 1.1 nM T54156 CWIM61 10364088 IC50 = 5150 nM T54156 CBA5I4 10365560 Ki = 0.8 nM T54156 C6WZ4F 10367355 IC50 = 30 nM T54156 C6FJU3 10367981 IC50 = 124 nM T54156 C8DJX4 10368307 Ki = 6 nM T54156 CJ96GA 10370197 IC50 = 74 nM T54156 CBTO07 10370226 Ki > 2128 nM T54156 C5VHS0 10370227 IC50 = 49 nM T54156 C6T4WO 10370281 Ki = 19 nM T54156 CUA47P 10371161 Ki = 2 nM T54156 C0IUQ7 10387351 Ki > 2128 nM T54156 CEM0U7 10387692 IC50 = 706 nM T54156 CL97HT 10388523 Ki = 77.75 nM T54156 CZNT94 10389113 IC50 = 5 nM T54156 CY2G0R 10391428 Ki > 2128 nM T54156 CR38WZ 10392467 IC50 = 11 nM T54156 C8UTS7 10393307 IC50 = 7.5 nM T54156 CFKA79 10395015 Ki > 2000 nM T54156 CTX2S3 10410319 Ki > 213 nM T54156 CRD6Z4 10410935 IC50 = 82 nM T54156 CZ90OC 10412486 Ki < 1 nM T54156 CA0TY8 10413076 Ki = 21 nM T54156 C98HMP 10413940 Ki = 288 nM T54156 CJ95UZ 10414150 IC50 = 57 nM T54156 C7K0HG 10414437 Ki = 691 nM T54156 CV4JT6 10415842 IC50 = 6.7 nM T54156 CZ3D4T 10428502 IC50 = 0.3 nM T54156 C31TIX 10428779 IC50 > 1000 nM T54156 CO6VM2 10436776 IC50 = 59 nM T54156 C7XE1L 10437629 IC50 = 90000 nM T54156 C9QS8N 10438212 IC50 = 2.1 nM T54156 C5WV1N 10439082 Ki > 2000 nM T54156 CA75GC 10453674 IC50 = 640 nM T54156 CQUR30 10454592 Ki = 0.41 nM T54156 C6T8VC 10456675 Ki = 0.6 nM T54156 CA5W6I 10458439 IC50 = 70 nM T54156 CP13CG 10459563 IC50 = 88 nM T54156 C8M9FE 10462640 Ki = 35600 nM T54156 CWV9Q2 10477531 Ki = 4.97 nM T54156 CHG02V 10478612 Ki = 3.68 nM T54156 CHL30D 10482442 IC50 = 75 nM T54156 CNQZ36 10483139 Ki = 1200 nM T54156 CA7HT2 10498521 Ki = 29 nM T54156 C6KD0A 10498747 IC50 = 0.9 nM T54156 CL8O6I 10500340 Ki = 120.23 nM T54156 CGK80V 10500816 Ki = 33 nM T54156 CVID65 10500886 Ki = 30.9 nM T54156 CP37WK 10501527 Ki = 25 nM T54156 CK6YN5 10501862 Ki = 7 nM T54156 C9QE1B 10502327 Ki = 7 nM T54156 CHOX65 10502351 IC50 = 16 nM T54156 CZ1R5Q 10502869 Ki = 6600 nM T54156 CO9S5H 10503708 Ki = 16 nM T54156 CT2NM3 10505241 Ki = 16 nM T54156 C65KOE 10506125 IC50 = 1900 nM T54156 C6D7JF 10506147 IC50 = 10000 nM T54156 CNH3L8 10506415 IC50 = 1320 nM T54156 C03MRW 10507152 Ki = 1.3 nM T54156 CDSO53 10507214 IC50 = 4.1 nM T54156 CC6H8T 10507755 Ki = 1 nM T54156 C9C5EL 10521197 IC50 = 5 nM T54156 CC2F5Y 10522311 IC50 = 1.8 nM T54156 CXD8I5 10523292 Ki = 125 nM T54156 CZ36JW 10523383 IC50 = 100000 nM T54156 C90HBF 10523728 Ki = 9 nM T54156 CX6EB7 10524337 Ki = 4500 nM T54156 CQTF46 10524338 Ki = 270 nM T54156 COT07L 10525329 IC50 = 7.6 nM T54156 C61GSD 10525562 IC50 = 1.6 nM T54156 CYB53K 10525912 Ki = 50 nM T54156 C56YKL 10525916 IC50 = 1200 nM T54156 C14XUW 10526101 IC50 = 3 nM T54156 CSLO13 10526877 IC50 = 7800 nM T54156 CEK90M 10527263 IC50 = 240 nM T54156 CA83ON 10527749 IC50 = 260 nM T54156 CJ0D7G 10528505 IC50 = 2.4 nM T54156 CBV6X5 10529587 IC50 = 2700 nM T54156 CGK37L 10529602 Ki = 1.995 nM T54156 CQ82VY 10530944 Ki = 25 nM T54156 CO2R0P 10544323 IC50 = 25 nM T54156 C0WHA9 10546565 Ki = 11 nM T54156 C06NQR 10547080 IC50 = 72 nM T54156 C40ZXE 10547784 Ki = 6 nM T54156 CS10ZB 10549106 Ki = 22 nM T54156 C4PK0U 10549114 IC50 = 3.7 nM T54156 C5JS8L 10549329 Ki = 1.288 nM T54156 CG27UI 10549756 Ki = 44 nM T54156 C2HJ1U 10549764 IC50 = 4.4 nM T54156 C82HQE 10550145 Ki = 8 nM T54156 CRHP20 10550304 IC50 = 1.8 nM T54156 C7WQ5Z 10550399 IC50 = 18 nM T54156 CNQ75F 10551139 IC50 = 17 nM T54156 C1FA6T 10551440 IC50 = 350 nM T54156 CCH0K3 10551483 IC50 = 3 nM T54156 C5UD0A 10551910 IC50 = 27000 nM T54156 CNE73L 10552476 IC50 = 28 nM T54156 C4K3UD 10552661 Ki = 13 nM T54156 CU8QP7 10552732 Ki = 10 nM T54156 CI8XG0 10554869 IC50 = 7700 nM T54156 CZ41HP 10554978 Ki = 23 nM T54156 CD3R8V 10562830 IC50 = 7.82 nM T54156 CT7O9M 10569678 IC50 = 3890.45 nM T54156 C8RWE4 10569743 IC50 = 19952.62 nM T54156 C0M4VN 10570699 IC50 = 40 nM T54156 CE14GM 10570702 IC50 = 2187.76 nM T54156 CUQ29Z 10571396 Ki = 100 nM T54156 C21VZS 10573362 IC50 = 0.2 nM T54156 C42IAF 10573603 Ki = 14 nM T54156 CG39CF 10574279 Ki = 9 nM T54156 C8LYR6 10574340 IC50 = 840 nM T54156 C42BTA 10576058 IC50 = 680 nM T54156 CH7Z2V 10576110 IC50 = 1700 nM T54156 C9YFC5 10577526 IC50 = 1500 nM T54156 CM4XT6 10578789 IC50 = 4300 nM T54156 CK05ZH 10579086 Ki = 0.5 nM T54156 C9L5OM 10579282 IC50 = 15.6 nM T54156 C3R2SO 10580533 Ki = 10 nM T54156 C8J6HS 10591505 Ki = 77.62 nM T54156 CB20LM 10594000 Ki = 41.69 nM T54156 CUTS47 10594564 IC50 = 58884.37 nM T54156 CN4Y6H 10594565 IC50 = 3800 nM T54156 CJQY74 10595685 IC50 = 2100 nM T54156 CI71CK 10595804 Ki = 11 nM T54156 CYNC76 10596158 IC50 = 9500 nM T54156 CD65NF 10597516 Ki = 39 nM T54156 CP2H8O 10597673 Ki = 8 nM T54156 CL7EX4 10598952 IC50 > 10000 nM T54156 CUZ73T 10599048 IC50 = 250 nM T54156 CN3E8J 10600844 Ki = 1.1 nM T54156 CJ86TP 10601066 IC50 = 8800 nM T54156 C6RH4O 10601640 IC50 = 13 nM T54156 CEJ1U0 10603377 Ki = 23 nM T54156 C5G9MI 10610114 Ki = 1700 nM T54156 CPW6A4 10617505 IC50 > 20000 nM T54156 CL02BO 10618584 IC50 = 16982.44 nM T54156 C06CAN 10619639 Ki = 14 nM T54156 CV14UH 10619971 Ki = 14 nM T54156 C8IZN2 10620836 IC50 = 87 nM T54156 CR69NK 10621302 IC50 = 340 nM T54156 CSQ96T 10621933 Ki = 0.76 nM T54156 CL5QN9 10622296 IC50 = 1.3 nM T54156 CVZ32G 10622447 Ki = 26 nM T54156 C4FYL1 10623748 IC50 = 16 nM T54156 C6R4EG 10624005 Ki = 5 nM T54156 CR8X1Q 10624346 IC50 = 8.2 nM T54156 CKF6D7 10625329 Ki = 3 nM T54156 CXV87K 10625636 IC50 = 1288.25 nM T54156 C98KGO 10625860 IC50 = 20 nM T54156 C70MFZ 10626445 Ki = 21 nM T54156 C5VGB1 10626732 Ki = 21 nM T54156 CL43CO 10627365 IC50 = 101 nM T54156 CA63VQ 10640307 Ki = 43 nM T54156 CPFH58 10641536 IC50 > 40000 nM T54156 CWRY91 10642128 IC50 = 2.3 nM T54156 CM1OZ6 10643325 IC50 = 14 nM T54156 C41RKE 10643401 Ki = 9 nM T54156 CUAI71 10643973 Ki = 1.4 nM T54156 CPYV83 10647658 Ki = 580 nM T54156 C2O1XM 10647817 IC50 = 4.1 nM T54156 CD96LY 10648089 Ki = 0.9 nM T54156 CVX7Q2 10648390 Ki = 14 nM T54156 CNF9I2 10648570 IC50 = 1288.25 nM T54156 C4TXZ1 10648776 Ki = 100 nM T54156 C5RWF4 10648802 IC50 = 2.1 nM T54156 C07FPQ 10649518 Ki = 69 nM T54156 COT6B8 10650624 Ki = 18 nM T54156 C69SPO 10650906 Ki = 1.2 nM T54156 CT23XW 10650907 Ki = 2.5 nM T54156 C27QHB 10663143 IC50 = 6.9 nM T54156 CGSX70 10664302 IC50 = 32.5 nM T54156 C97KZU 10665624 IC50 = 64000 nM T54156 CW1E7L 10667540 IC50 = 240 nM T54156 CF0E6H 10668745 IC50 = 19952.62 nM T54156 CSCL07 10668823 Ki = 7.9 nM T54156 CFYC35 10669215 Ki = 2.5 nM T54156 C6TC0Z 10669216 Ki = 2.8 nM T54156 C8HK0C 10669534 IC50 = 2.3 nM T54156 C78GYJ 10670529 IC50 = 5 nM T54156 CY6QC1 10670819 IC50 = 5 nM T54156 C5FWS1 10670820 IC50 = 24 nM T54156 C4QVL0 10670896 Ki = 5 nM T54156 CPG5O2 10671155 IC50 = 3.8 nM T54156 CB1F4G 10671203 IC50 = 580 nM T54156 C3DXN5 10671411 Ki = 1.7 nM T54156 CWB19K 10671441 Ki = 1.288 nM T54156 C09LJR 10671827 IC50 = 6.6 nM T54156 CXDM24 10671863 Ki = 0.68 nM T54156 CU5M1J 10691797 Ki = 18 nM T54156 CR5KF8 10692994 IC50 = 100000 nM T54156 C8JX1G 10693698 Ki = 7 nM T54156 CM1T7K 10694510 Ki = 3 nM T54156 C7SM1E 10694604 Ki = 8.7 nM T54156 C3E1DX 10695165 IC50 = 12 nM T54156 C7ZQM4 10695491 Ki = 1.5 nM T54156 C6MWX8 10696713 IC50 = 22 nM T54156 CG5JM9 10698412 Ki = 3 nM T54156 C56VSE 10698786 Ki = 1.6 nM T54156 C5E8QF 10707457 Ki = 137 nM T54156 C78CKH 10715629 IC50 > 20000 nM T54156 C0ZX6T 10717308 IC50 = 4900 nM T54156 C3TGW8 10717400 Ki = 36 nM T54156 CZ1M3L 10718058 Ki = 13 nM T54156 CQZ7M8 10718133 Ki = 21 nM T54156 CI64YZ 10718883 IC50 = 3.6 nM T54156 CB96HF 10718916 IC50 > 10000 nM T54156 CVPC97 10718960 IC50 = 570 nM T54156 CN8AK6 10718996 Ki = 0.78 nM T54156 C2IS9D 10719476 Ki = 1.4 nM T54156 CF46SQ 10721337 Ki = 22 nM T54156 CC1FB8 10721904 Ki = 3.1 nM T54156 CB2QD0 10723468 Ki = 1.3 nM T54156 C8KE2C 10735676 IC50 = 2900 nM T54156 CO7VP4 10737552 Ki = 15 nM T54156 C51DZG 10737732 IC50 = 16000 nM T54156 C1LS5U 10738104 IC50 = 27 nM T54156 C76ANK 10739335 IC50 = 0.6 nM T54156 CB8G2D 10739728 Ki = 17 nM T54156 C0T2VK 10740460 IC50 = 1.7 nM T54156 C4FWC9 10740485 Ki = 120 nM T54156 CKJD45 10741133 IC50 = 84000 nM T54156 C0WKL7 10741470 Ki = 17 nM T54156 CPDX27 10741484 IC50 > 10000 nM T54156 C0QT2F 10741956 Ki = 7 nM T54156 CLI7B3 10742101 IC50 > 10000 nM T54156 C39DPG 10742191 IC50 = 28 nM T54156 CY2BZ0 10742536 Ki = 53 nM T54156 CCH94Q 10743507 IC50 = 1.2 nM T54156 CTA0Y4 10743933 IC50 = 1200 nM T54156 C5BZ0J 10745489 Ki = 29 nM T54156 C9ILP3 10745718 IC50 = 10000 nM T54156 CK30AE 10745748 Ki = 0.7 nM T54156 CWF50D 10745851 Ki = 36 nM T54156 CA3F1N 10758013 Ki = 100 nM T54156 CY9W4M 10760229 IC50 = 1100 nM T54156 CDX13Z 10761730 Ki = 10 nM T54156 CA4U7D 10762262 Ki = 16 nM T54156 CP2G0N 10763745 Ki = 1.7 nM T54156 CJG14B 10764335 IC50 = 870 nM T54156 CM54WS 10764477 Ki = 9800 nM T54156 C0ZJB9 10764600 IC50 = 32 nM T54156 CY8LV5 10765345 IC50 = 210 nM T54156 COAL70 10765803 IC50 = 52 nM T54156 CA6C0Z 10766622 Ki = 1.096 nM T54156 C0R1ZA 10767025 Ki = 3.7 nM T54156 CNT4D0 10767387 Ki = 30 nM T54156 CN83AJ 10768085 IC50 = 2600 nM T54156 C01YKA 10768236 IC50 = 17 nM T54156 CQ6U2Y 10780743 Ki = 30 nM T54156 C15PVT 10785952 Ki = 27 nM T54156 CLAP90 10785969 IC50 = 40 nM T54156 C8AF9L 10787938 Ki = 1.2 nM T54156 CNAE08 10788733 IC50 = 4900 nM T54156 CKV2O8 10789493 IC50 = 0.6 nM T54156 CM74LH 10789594 IC50 = 5.9 nM T54156 C9NZ4W 10789711 IC50 = 1.9 nM T54156 C0NP2Z 10790811 IC50 > 10000 nM T54156 C31EHR 10791372 IC50 = 23 nM T54156 C3P7LZ 10792025 Ki = 3.981 nM T54156 C8D1EN 10792133 IC50 = 2000 nM T54156 C6FWC1 10808125 IC50 = 0.9 nM T54156 C5HF8Z 10809178 IC50 = 400 nM T54156 CP72JG 10810483 IC50 = 4.4 nM T54156 CU9F7V 10810684 Ki = 38.9 nM T54156 CS0O7M 10811110 Ki = 42 nM T54156 C49HCM 10812120 IC50 = 270 nM T54156 CV3ZA5 10812444 IC50 = 8.3 nM T54156 CEM1J0 10812918 IC50 = 60 nM T54156 CUOB87 10816515 Ki = 1.1 nM T54156 C34KQG 10816626 IC50 = 3200 nM T54156 CS7BY4 10816934 IC50 = 4800 nM T54156 CBL54W 10816989 IC50 = 4400 nM T54156 C3AI5Z 10831752 IC50 = 65000 nM T54156 CMX2J7 10832371 IC50 > 50000 nM T54156 CF50HD 10832925 IC50 = 6700 nM T54156 COE82D 10833334 Ki = 122 nM T54156 C5OG4U 10833497 IC50 = 38000 nM T54156 C2A0IX 10833840 IC50 = 11 nM T54156 C9M1JI 10834357 Ki = 26.92 nM T54156 CND0X1 10834889 IC50 = 110 nM T54156 C48PYQ 10836923 IC50 = 2.6 nM T54156 CT3MN0 10837022 Ki = 7.1 nM T54156 CGR16B 10837261 IC50 = 1100 nM T54156 CR0E9Q 10837740 Ki = 5 nM T54156 C9H4CP 10838922 Ki = 1.1 nM T54156 CB32OK 10838949 IC50 = 1500 nM T54156 CR50UM 10839419 Ki = 7 nM T54156 CL1KG7 10840630 Ki = 28 nM T54156 C6ZSP8 10862104 Ki = 3.6 nM T54156 CQ1L7C 10863755 Ki > 2128 nM T54156 CF72UK 10864417 IC50 = 8.5 nM T54156 C6CD3R 10873386 Ki = 1.1 nM T54156 C0AQL8 10873958 Ki = 7 nM T54156 CBQ70P 10874312 IC50 = 3 nM T54156 CLG40T 10874819 IC50 = 2.3 nM T54156 CXY47P 10875332 IC50 = 132 nM T54156 CXGN38 10875470 IC50 = 190 nM T54156 CJ0LE4 10876254 Ki = 183 nM T54156 CIB8Y1 10884337 Ki = 19 nM T54156 C3AY8O 10885569 IC50 = 31 nM T54156 CAU0I3 10885834 IC50 = 13.9 nM T54156 CG1I4Y 10886343 IC50 = 2 nM T54156 CF5L1R 10886549 IC50 = 7 nM T54156 CA64PN 10886607 IC50 = 43 nM T54156 CDZ04P 10887027 Ki = 91 nM T54156 C0R5QL 10894433 Ki = 5.05 nM T54156 C7AMS4 10895808 Ki = 1209 nM T54156 C1M8OI 10896082 Ki = 5.2 nM T54156 CPJ0I8 10896934 IC50 = 39 nM T54156 CU7YE0 10896986 IC50 = 0.2 nM T54156 CMV89R 10897017 IC50 = 48 nM T54156 C3FQT7 10903871 Ki = 35 nM T54156 CX93MR 10907320 IC50 = 30 nM T54156 CM9G8A 10907701 IC50 = 2 nM T54156 CSK87I 10907725 IC50 = 22 nM T54156 C13CJH 10907740 IC50 = 37 nM T54156 C69ZTR 10913644 Ki = 1050 nM T54156 C2QR0W 10914151 Ki = 586 nM T54156 CAH70N 10914350 IC50 = 49 nM T54156 CF9NT3 10914471 IC50 = 447 nM T54156 C2M4PK 10916140 Ki = 349 nM T54156 C7XE3L 10917417 Ki < 2.1 nM T54156 C6L7WH 10927616 Ki = 10.99 nM T54156 CGI2T1 10928606 IC50 = 341 nM T54156 CXHA75 10928874 IC50 = 94.9 nM T54156 C40PRC 10929100 IC50 = 15 nM T54156 CXY4L6 10929354 IC50 = 661 nM T54156 CDSQ41 10929404 IC50 = 24 nM T54156 CLIR35 10938505 IC50 = 2 nM T54156 C1QVT6 10939850 IC50 = 3.9 nM T54156 CWO29J 10940364 IC50 = 35 nM T54156 CL64UM 10940712 IC50 = 12 nM T54156 C89IYC 10948209 Ki < 2.1 nM T54156 C7GH8P 10948665 Ki = 12.8 nM T54156 C2TA9N 10949166 Ki = 5.05 nM T54156 C5C4KV 10949301 Ki = 3.802 nM T54156 CC46WL 10950008 Ki > 2000 nM T54156 C9YOU4 10951375 IC50 = 4.3 nM T54156 CJI1G0 10951750 IC50 = 0.2 nM T54156 CNBR78 10952384 IC50 = 1.88 nM T54156 C0A2IR 10958121 Ki = 11 nM T54156 C3K1BL 10959017 IC50 = 11 nM T54156 C7PX8G 10960109 Ki > 800 nM T54156 C5HS4F 10961382 Ki > 2128 nM T54156 CMY8S6 10961569 IC50 = 0.9 nM T54156 CPA1Q2 10961828 IC50 = 4.9 nM T54156 C5ZV9Q 10962137 IC50 = 58 nM T54156 CJU03W 10969502 Ki = 316.23 nM T54156 C30FBA 10970628 Ki = 29 nM T54156 CQ68IE 10972732 IC50 = 4.1 nM T54156 CJHO94 10972891 IC50 = 2.2 nM T54156 CTP6I0 10973485 IC50 = 9.7 nM T54156 C9DM0P 10980832 Ki = 80 nM T54156 CL7K8S 10983560 Ki < 1 nM T54156 C3UH2B 10983665 Ki = 981 nM T54156 CR9J5B 10983887 IC50 = 3.8 nM T54156 C68LPK 10983913 IC50 = 1.8 nM T54156 CJ8I9G 10983916 IC50 = 19 nM T54156 CS7D0Z 10984030 IC50 = 1.4 nM T54156 CV4J2F 10984597 IC50 = 0.01 nM T54156 C0NIX9 10985227 IC50 = 379 nM T54156 C0G8TE 10993343 Ki = 40 nM T54156 CW8Z6R 10993677 Ki = 2128 nM T54156 CCX0L6 10994350 IC50 = 1 nM T54156 CW0Y6I 10994897 IC50 = 6.2 nM T54156 CA5I7L 10995373 IC50 = 35 nM T54156 C9C8SA 11001101 IC50 = 128 nM T54156 C3QX0T 11005761 IC50 = 10 nM T54156 CMN17S 11005934 IC50 = 0.34 nM T54156 CJM41O 11006091 IC50 = 2 nM T54156 C4PNK3 11006191 IC50 = 149 nM T54156 C95NXQ 11006894 Ki = 21 nM T54156 C7WEZ4 11009332 Ki = 34000 nM T54156 CS4FL3 11012667 IC50 = 141 nM T54156 C5JE9G 11014504 IC50 = 197 nM T54156 C8ERT5 11014626 Ki > 800 nM T54156 C75DGS 11015731 Ki = 358 nM T54156 C9WPH7 11016072 Ki = 200 nM T54156 CBE68H 11016073 Ki > 15000 nM T54156 CG2DK0 11016448 IC50 = 11.7 nM T54156 C3IYK8 11016511 IC50 = 0.96 nM T54156 CF30UR 11016519 IC50 = 3.2 nM T54156 CODQ51 11016616 IC50 = 6.6 nM T54156 CO6C8A 11017232 IC50 = 115 nM T54156 CM1H5P 11026185 Ki = 2.1 nM T54156 CQD70Y 11026301 Ki = 483 nM T54156 C6IHF5 11026991 IC50 > 6 nM T54156 C3LF1Y 11027584 Ki > 2128 nM T54156 CF5KU1 11027718 IC50 = 5.5 nM T54156 CA49QF 11027968 IC50 = 1.4 nM T54156 CLXZ15 11037377 Ki = 3.2 nM T54156 C0ERN9 11037836 Ki = 411 nM T54156 CT2S0G 11038175 IC50 = 4.1 nM T54156 C83AKP 11038896 IC50 = 51 nM T54156 CG3B5N 11039339 IC50 = 49 nM T54156 C3W9IT 11046880 Ki = 166 nM T54156 CZO40T 11048604 Ki > 800 nM T54156 C5R7JX 11049650 Ki > 2128 nM T54156 CW42KO 11049937 IC50 = 2 nM T54156 C23KPN 11050468 IC50 = 0.5 nM T54156 C9RU4I 11059620 IC50 = 176.5 nM T54156 CH8O1E 11060081 Ki > 2128 nM T54156 CM6X1E 11061555 Ki > 2000 nM T54156 C49PNL 11069047 Ki = 3.6 nM T54156 C1N5PT 11070986 IC50 = 137 nM T54156 C18EIZ 11071831 IC50 = 9.1 nM T54156 C2LSU0 11072397 IC50 = 71 nM T54156 C5MUD2 11078779 IC50 = 71 nM T54156 C43JOG 11080156 Ki = 39 nM T54156 CT3VX4 11080936 Ki = 2128 nM T54156 CG0A4C 11081333 IC50 = 37 nM T54156 CVJX34 11081788 Ki < 1 nM T54156 C05MUK 11081992 IC50 = 0.5 nM T54156 C6XI8J 11082293 IC50 = 11 nM T54156 CUNM68 11083152 Ki > 2128 nM T54156 CF0NJ9 11090097 IC50 = 0.14 nM T54156 CS29GX 11091928 IC50 = 3.8 nM T54156 C16WBE 11092175 IC50 = 19 nM T54156 CE8V9B 11092295 IC50 = 0.9 nM T54156 CR8ZA7 11092551 IC50 = 16 nM T54156 CT2CH7 11092701 IC50 = 12 nM T54156 C6R7XB 11092861 Ki > 2128 nM T54156 CWT6C7 11092884 IC50 = 55 nM T54156 CX69YN 11093502 IC50 = 0.3 nM T54156 C6CLV8 11101735 IC50 = 2930 nM T54156 CR4V2D 11101785 Ki = 160 nM T54156 C8CK3E 11102531 IC50 = 76 nM T54156 C57OXT 11102540 Ki = 4.46 nM T54156 CA2OS3 11103408 IC50 = 13 nM T54156 C6G2DI 11111616 Ki = 3 nM T54156 CUK03P 11112062 Ki = 1634 nM T54156 CWV45Z 11112302 Ki < 2.1 nM T54156 CEAI92 11112993 IC50 = 3 nM T54156 CY1SR9 11113744 IC50 = 597 nM T54156 CI1GS5 11114351 IC50 = 602 nM T54156 CUO7B3 11122933 Ki = 3.3 nM T54156 CNGP50 11122963 IC50 = 0.26 nM T54156 CB2I5K 11123701 IC50 = 23 nM T54156 C8YVE5 11123989 IC50 = 4 nM T54156 C3PR1J 11124862 IC50 = 89 nM T54156 CAJ27B 11124943 IC50 = 22 nM T54156 CNBG53 11124956 IC50 = 0.6 nM T54156 CX2B6C 11125147 Ki = 1170 nM T54156 C9GJ7C 11133809 Ki = 993 nM T54156 C2YBQ7 11134935 IC50 = 71.5 nM T54156 C8DMW5 11135133 IC50 = 512 nM T54156 CD3N8B 11135304 IC50 = 29 nM T54156 CPO02F 11142863 IC50 = 9.2 nM T54156 CF52TX 11143173 Ki = 3324 nM T54156 C3V4ZX 11143285 IC50 = 16 nM T54156 CH61QF 11144824 IC50 = 0.9 nM T54156 C8HM2R 11145437 Ki = 347 nM T54156 CHF19X 11146467 Ki = 118 nM T54156 C5WS3E 11147931 IC50 = 2000 nM T54156 CM0QK6 11156328 IC50 = 14 nM T54156 CZ8KI2 11157757 IC50 = 550 nM T54156 CVI3F8 11188429 IC50 > 10000 nM T54156 C2LZ7F 11191803 IC50 = 26 nM T54156 CCQ6N8 11194666 IC50 > 100000 nM T54156 CO5VN2 11201367 IC50 > 10000 nM T54156 CO76XI 11205873 IC50 = 3000 nM T54156 C9R7OM 11207122 IC50 > 100000 nM T54156 C3LEA2 11226622 IC50 = 2 nM T54156 C72UCB 11233687 IC50 = 124 nM T54156 CPV9L7 11246575 Ki = 14 nM T54156 CUOH67 11252195 IC50 > 100000 nM T54156 CJZ3P6 11257884 Ki = 0.87 nM T54156 CD1FT8 11258906 IC50 = 18 nM T54156 CO7T3M 11261246 IC50 = 16 nM T54156 CC62RY 11279665 IC50 = 11 nM T54156 CF9O2R 11286824 IC50 > 100000 nM T54156 C1IW7N 11292680 IC50 = 6.7 nM T54156 C8C5AV 11294179 Ki > 2128 nM T54156 C7H9JG 11295013 IC50 = 1 nM T54156 C78QSH 11307739 IC50 = 57 nM T54156 CJ09XO 11317090 IC50 = 2 nM T54156 CK91YW 11317404 IC50 = 2500 nM T54156 CJ5SU9 11328354 Ki > 300000 nM T54156 CN2P4G 11328571 IC50 = 1876 nM T54156 CQH57S 11342435 IC50 > 7000 nM T54156 CZ8B0D 11349945 Ki < 2.1 nM T54156 CCKI02 11360440 Ki = 2 nM T54156 C7QNX8 11363138 IC50 > 5000 nM T54156 CM8Y1J 11367571 IC50 > 100000 nM T54156 CTQK48 11373358 Ki > 2128 nM T54156 C48DYJ 11374008 Ki = 7.4 nM T54156 CL8QO7 11382562 IC50 = 1500 nM T54156 CNZ0T5 11386918 IC50 = 10 nM T54156 COZN84 11388372 IC50 = 20 nM T54156 CUJ4V0 11391937 IC50 = 7.28 nM T54156 C13NCF 11400989 IC50 = 20000 nM T54156 C3EX5J 11407165 Ki = 47 nM T54156 CZM5E8 11410471 IC50 = 26 nM T54156 C2EUO5 11417011 IC50 > 10000 nM T54156 CK95HW 11429232 Ki = 0.9 nM T54156 C01FLQ 11441438 Ki = 8.5 nM T54156 CZY3W9 11444262 IC50 = 19 nM T54156 CI0V6L 11447356 IC50 > 100000 nM T54156 C5NAJ3 11449819 IC50 = 186 nM T54156 CCMT46 11457732 IC50 > 100000 nM T54156 C96DRO 11466734 IC50 = 24000 nM T54156 C7QF0G 11467517 IC50 = 12000 nM T54156 CQ1D6E 11470070 IC50 = 1000 nM T54156 C1KP2Q 11473879 Ki > 2128 nM T54156 C5QEZ8 11483818 IC50 = 148 nM T54156 C5G8PM 11511807 IC50 > 5000 nM T54156 C1NZB9 11548265 IC50 = 9 nM T54156 CIWP38 11555036 IC50 = 22 nM T54156 C3H2DG 11577137 IC50 = 100 nM T54156 CXT05D 11581283 IC50 = 3390 nM T54156 CUL5H2 11605631 IC50 = 25 nM T54156 CXKU59 11620780 IC50 > 5000 nM T54156 CCBS59 11634234 IC50 = 1670 nM T54156 CZO71U 11639846 IC50 = 1510 nM T54156 CFV49P 11641262 IC50 < 1.5 nM T54156 CR2UN0 11669859 IC50 = 19.5 nM T54156 CK9F4P 11673778 IC50 = 14000 nM T54156 C90GCV 11675055 IC50 = 9290 nM T54156 C28WNK 11682752 Ki = 180 nM T54156 CKGR97 11692294 IC50 > 5000 nM T54156 C1MJ3P 11713694 IC50 = 535 nM T54156 C2BJ3X 11716217 Ki = 100000 nM T54156 C4FU2H 11717997 IC50 = 10030 nM T54156 C4ECU2 11720597 IC50 = 955 nM T54156 C4CKB0 11725943 IC50 = 13000 nM T54156 CCD93H 11730086 Ki = 90 nM T54156 CBT48P 11731926 Ki = 7 nM T54156 CA43HK 11732287 Ki = 10.5 nM T54156 C68KBY 11732585 Ki = 96 nM T54156 C7CED0 11733417 IC50 = 2990 nM T54156 CI0KL2 11733573 IC50 = 24 nM T54156 C64LQC 11733862 Ki > 2000 nM T54156 C27SBC 11734162 IC50 = 1 nM T54156 CIU03K 11734219 Ki > 2128 nM T54156 CJOE40 11748355 Ki = 9 nM T54156 C4HD9K 11751106 IC50 = 1443 nM T54156 CO8QT0 11753905 Ki = 1720 nM T54156 C3P0TZ 11754739 Ki = 5800 nM T54156 CJ4G5D 11754907 IC50 = 3.6 nM T54156 CE6OS0 11755521 IC50 = 1.2 nM T54156 CD6S0B 11757331 IC50 = 26080 nM T54156 C5E7KU 11757592 Ki = 0.9 nM T54156 CUC9R5 11758082 IC50 = 0.2 nM T54156 CZ5V9G 11758096 IC50 = 3.8 nM T54156 C2KU3D 11760296 IC50 = 51 nM T54156 C3RW1X 11761191 Ki = 3.9 nM T54156 CQ3Y4E 11761293 IC50 = 200 nM T54156 C6K8HR 11761578 Ki > 2128 nM T54156 CE1HZ4 11761760 Ki < 1 nM T54156 CQP12F 11787159 IC50 = 10 nM T54156 C7BV5P 11792968 Ki = 89 nM T54156 CV16JZ 11793588 IC50 = 1200 nM T54156 CKM6P2 11795228 IC50 = 17 nM T54156 CCSD72 11795621 IC50 = 3.6 nM T54156 CY8N1U 11795715 Ki = 3 nM T54156 CY7H2T 11795824 Ki = 8 nM T54156 C3DE6J 11796352 IC50 = 210 nM T54156 CK24XT 11796481 Ki = 12 nM T54156 CHB01Z 11797196 IC50 = 1700 nM T54156 CJ4VL3 11797382 IC50 = 61 nM T54156 CKUM64 11797718 IC50 = 1180 nM T54156 C7VLP9 11798303 IC50 = 86 nM T54156 CZ3C9P 11798873 IC50 = 7.3 nM T54156 C19RCP 11799753 Ki = 4.571 nM T54156 CZ5LP1 11800650 IC50 = 2300 nM T54156 C2YD4N 11809525 IC50 = 35 nM T54156 C1NRV6 11811437 IC50 = 8 nM T54156 CQ9HE2 11811551 IC50 = 1760 nM T54156 CSG07A 11811629 Ki > 800 nM T54156 CK03NI 11811717 Ki = 66 nM T54156 CLW3F1 11812791 IC50 = 415 nM T54156 C20PYA 11813392 IC50 = 1.7 nM T54156 CH3SV6 11813493 IC50 = 47 nM T54156 CZ08ID 11814382 IC50 = 143 nM T54156 C8DY3Z 11817193 IC50 > 100000 nM T54156 CEN02U 11822212 Ki = 567 nM T54156 CDU9S2 11824087 Ki = 751 nM T54156 C7BK5P 11825105 IC50 = 0.5 nM T54156 CKEM29 11827006 IC50 = 12 nM T54156 CV2MX4 11832221 Ki = 242 nM T54156 C48QEH 11833533 Ki = 100 nM T54156 C02BWA 11967143 Ki > 2000 nM T54156 CB80OT 12000718 IC50 > 20000 nM T54156 C43PJZ 12000720 IC50 > 20000 nM T54156 CJ3HA6 12443210 IC50 = 50000 nM T54156 C0JID3 12447203 Ki > 100000 nM T54156 CTHQ39 12635073 Ki = 12000 nM T54156 CIQX87 12635074 Ki = 73000 nM T54156 C0XKJ1 12671872 IC50 > 100000 nM T54156 CSR94V 13559594 IC50 = 2.35 nM T54156 C71ASU 13644537 IC50 = 7.25 nM T54156 CQTX49 13738810 IC50 > 100000 nM T54156 C1AJO7 13968141 IC50 > 300000 nM T54156 CM9PD5 14237653 IC50 = 27300 nM T54156 CA2H8V 14303060 IC50 = 150 nM T54156 C1IZ7D 15296597 Ki = 34.67 nM T54156 CGH19T 15296844 IC50 > 300000 nM T54156 CSU04W 15406874 IC50 = 230 nM T54156 CKN3R1 15430588 IC50 = 318 nM T54156 C63MFQ 15435266 IC50 = 5 nM T54156 COZM90 15485452 IC50 = 0.14 nM T54156 CEM2O0 15485453 IC50 = 250 nM T54156 CP2C4Z 15524387 Ki = 21200 nM T54156 CAF7R5 15524388 Ki = 203 nM T54156 C17HGN 15524389 Ki = 15500 nM T54156 CFH8Y6 15524390 Ki = 22000 nM T54156 CU7CM3 15551877 IC50 = 7 nM T54156 C3N1KV 15629940 IC50 > 100000 nM T54156 C5TLB4 15765753 IC50 = 4.25 nM T54156 C2WHJ4 15859211 IC50 = 650 nM T54156 C5FA3L 15871222 IC50 < 0.1 nM T54156 CB3A4Z 15941413 Ki = 390 nM T54156 CA40FE 15941550 Ki = 160 nM T54156 CM3D1L 15941553 Ki = 130 nM T54156 CQ0ZL7 15941677 Ki = 5 nM T54156 C6F9WV 15941679 Ki = 330 nM T54156 C7C1HI 15941680 Ki = 520 nM T54156 C6R1LD 15985818 IC50 = 777 nM T54156 CV67UL 15986261 IC50 = 23000 nM T54156 CU2C1R 15987326 IC50 > 10000 nM T54156 C4WX2I 16108938 IC50 > 5000 nM T54156 CD51GI 16108939 IC50 = 113 nM T54156 C5YVB0 16108940 IC50 > 5000 nM T54156 CB4DU9 16108941 IC50 > 5000 nM T54156 CBW71J 16108942 IC50 > 5000 nM T54156 CG6R9L 16108943 IC50 > 3000 nM T54156 CN62KM 16108944 IC50 > 5000 nM T54156 C7YS5Q 16108947 IC50 = 650 nM T54156 CLD2Y4 16108948 IC50 > 5000 nM T54156 CJR95O 16108949 IC50 > 5000 nM T54156 CRQ26L 16108950 IC50 > 5000 nM T54156 CH80AG 16108951 IC50 = 77 nM T54156 CWB0G9 16108952 IC50 > 5000 nM T54156 CS46XU 16126723 IC50 = 3.2 nM T54156 CC6OH2 16129741 IC50 = 39200 nM T54156 CYHI93 16418978 IC50 = 44200 nM T54156 CH7D2Q 16420684 IC50 = 13000 nM T54156 C91EXN 16655061 IC50 = 920 nM T54156 CQS0F5 16719301 IC50 > 10000 nM T54156 C75XDI 16730519 IC50 > 2000 nM T54156 C3S2TQ 17754305 IC50 = 1010 nM T54156 CIR7S8 17866387 IC50 = 2 nM T54156 CL1H9W 17866459 IC50 = 7 nM T54156 C9RNH3 17866675 IC50 = 1 nM T54156 CCGR13 17897285 IC50 = 9 nM T54156 C2ZAX1 18002715 Ki > 2100 nM T54156 C12UGK 18002722 Ki > 2100 nM T54156 C0IYW8 18002726 Ki > 2100 nM T54156 C8N1DM 18002729 Ki > 2100 nM T54156 CCG96A 18002736 Ki > 2100 nM T54156 C5MLG1 18002745 Ki > 2100 nM T54156 CXT4H2 18002752 Ki > 2100 nM T54156 C26WHK 18002758 Ki > 2100 nM T54156 CV90XS 18002764 Ki > 2100 nM T54156 C8KPM7 18002765 Ki > 2100 nM T54156 CMJ0K3 18002771 Ki > 2100 nM T54156 C2CO9Z 18002775 Ki > 2100 nM T54156 CK8FS7 18173159 IC50 = 33 nM T54156 CX10BM 18173179 IC50 = 25 nM T54156 CQO70Y 18173222 IC50 = 221 nM T54156 CI53DY 18379040 Ki > 2128 nM T54156 CB1U5T 18379077 Ki > 2128 nM T54156 CSX97G 18379115 Ki > 2128 nM T54156 CJHL25 18379123 Ki > 2128 nM T54156 CR0B8G 18379149 Ki > 2128 nM T54156 CS4V5K 18379187 Ki > 2128 nM T54156 CCTY94 18379210 Ki > 2128 nM T54156 CA6K5S 18379235 Ki > 2128 nM T54156 CCSK49 18379254 Ki > 2128 nM T54156 CP4T7S 18379435 Ki > 2128 nM T54156 C9Y5GX 18379443 Ki > 2128 nM T54156 CSY0N8 18394511 IC50 > 300000 nM T54156 CO21QH 18395616 IC50 = 6 nM T54156 C5B9WG 18533077 IC50 = 400 nM T54156 C50AEZ 18616892 IC50 = 450 nM T54156 CIEH93 19382975 IC50 = 6000 nM T54156 C60WKH 20196702 IC50 = 5.28 nM T54156 CK8MP3 20620240 Ki = 160 nM T54156 CPC4G6 20620273 Ki = 370 nM T54156 C2E3CY 20620614 IC50 = 1100 nM T54156 CV1SD8 20620714 IC50 = 180 nM T54156 C3GAC4 20620715 IC50 = 380 nM T54156 C5RQ8A 20620860 IC50 = 960 nM T54156 CA7FK0 20639531 IC50 = 31 nM T54156 CMX23W 20639537 IC50 = 1 nM T54156 C34XRP 20639540 IC50 = 3 nM T54156 C7AP8Z 20639546 IC50 = 30 nM T54156 CPK09X 20651316 IC50 = 0.9 nM T54156 CG1BD4 20689551 IC50 = 1200 nM T54156 C48TWB 20728102 IC50 > 2000 nM T54156 C18RXS 20735191 IC50 = 0.1 nM T54156 C4I1OM 20735209 IC50 = 1230 nM T54156 CW3D7O 20760308 Ki = 366 nM T54156 CA7JE6 20924268 IC50 = 25000 nM T54156 CG18HB 21310751 IC50 = 11 nM T54156 CEW0M3 21310753 IC50 = 3 nM T54156 CC2L1Z 21310756 IC50 = 554 nM T54156 CWM7F2 21310775 IC50 = 23 nM T54156 CNEW70 21310777 IC50 = 22.91 nM T54156 CY12PI 21310778 IC50 = 12.88 nM T54156 CV10FJ 21310779 IC50 = 27 nM T54156 CPT4E5 21310780 IC50 = 346 nM T54156 CJ2U7K 21310781 IC50 = 353 nM T54156 C5SG2L 21310789 IC50 = 8 nM T54156 C3TI6Y 21310790 IC50 = 8 nM T54156 C87BMF 21310824 IC50 = 5 nM T54156 C26IPQ 21310829 IC50 = 15 nM T54156 CIB1X5 21310851 IC50 = 10 nM T54156 C6OZL3 21310926 IC50 = 5 nM T54156 C72BVA 21310934 IC50 = 440 nM T54156 CUJ6A1 21310984 IC50 = 144 nM T54156 CAS84B 22004289 Ki = 230 nM T54156 C1MCG7 22004293 Ki = 39 nM T54156 CH6U1G 22338710 IC50 = 46 nM T54156 CO91AD 22341241 Ki > 2128 nM T54156 CE5DH1 22484408 IC50 = 500 nM T54156 CZT05X 22484417 Ki > 10000 nM T54156 CZT64B 22484431 Ki = 1600 nM T54156 CAM10T 22485252 IC50 = 42.5 nM T54156 CBJS34 22485260 IC50 < 0.1 nM T54156 C9MU7N 22485263 IC50 = 265 nM T54156 CEGJ03 22485276 IC50 = 82.3 nM T54156 C7VB8G 22485289 IC50 < 0.1 nM T54156 CNB02I 22485291 IC50 < 0.1 nM T54156 CAY3N6 22485292 IC50 = 2.2 nM T54156 C94OCJ 22485302 IC50 = 0.2 nM T54156 C3YL5X 22485311 IC50 = 2 nM T54156 CWA03L 22485327 IC50 = 1.1 nM T54156 C6JRW5 22485340 IC50 = 0.21 nM T54156 C5JZF1 22485344 IC50 = 5 nM T54156 CI7MY5 22485346 IC50 = 1.7 nM T54156 CI1YL7 22485347 IC50 = 0.27 nM T54156 C25OBD 22485356 IC50 = 2.9 nM T54156 C7I0EW 22485367 IC50 < 0.1 nM T54156 CL64TJ 22485368 IC50 = 1.5 nM T54156 CT4GF9 22485381 IC50 > 10000 nM T54156 C27NDB 22485386 IC50 = 4 nM T54156 C3MG9P 22485396 IC50 = 3.8 nM T54156 CZY10U 22485408 IC50 = 1.9 nM T54156 C89AGT 22485413 IC50 = 0.3 nM T54156 C03NLM 22485417 IC50 = 0.4 nM T54156 C8GHU9 22485432 IC50 = 1.9 nM T54156 C0K1GE 22645081 IC50 = 40 nM T54156 C2Q4XK 22707806 IC50 = 0.1 nM T54156 CVF9M4 22922043 IC50 = 14280 nM T54156 COCN69 22956916 Ki = 767 nM T54156 C85PXN 22956934 Ki = 252 nM T54156 CIYA45 22985930 IC50 = 0.22 nM T54156 CF75MS 23017979 IC50 = 53000 nM T54156 CQJ3S4 23018008 IC50 = 28000 nM T54156 C4VG8C 23506747 IC50 = 455 nM T54156 CK97AT 23506779 IC50 = 21 nM T54156 CP94QR 23506783 IC50 = 11 nM T54156 C6IZ1S 23513821 IC50 = 879 nM T54156 CPNM93 23513825 IC50 = 454 nM T54156 CML90Q 23513831 IC50 = 972 nM T54156 CD3U8A 23627203 Ki = 6300 nM T54156 C8UIC6 23644662 Ki > 100000 nM T54156 CCLA40 23644663 Ki > 100000 nM T54156 CSZ6J4 23645528 Ki = 4.266 nM T54156 C6UH9Q 23645529 Ki = 1.4 nM T54156 CD0JP3 23645530 Ki = 1.2 nM T54156 CM37EC 23645531 Ki = 4.266 nM T54156 C9PD5F 23645532 Ki = 4.365 nM T54156 C1OE7R 23645533 Ki = 1 nM T54156 CCSN04 23645534 Ki = 1.5 nM T54156 CU08WI 23645535 Ki = 0.6 nM T54156 CY41UC 23645536 Ki = 28 nM T54156 CX15EH 23645537 Ki = 5 nM T54156 CD3Q6G 23645538 Ki = 30.9 nM T54156 CE6NQ2 23645539 Ki = 21000 nM T54156 C4VK3U 23645540 Ki = 21000 nM T54156 C8VM1C 23645541 Ki = 83000 nM T54156 C0MUT6 23645542 Ki = 14000 nM T54156 CNI07H 23645543 Ki = 13000 nM T54156 CHK2X1 23645544 Ki = 23000 nM T54156 CW1V2Z 23645545 Ki = 13000 nM T54156 C6SP7T 23645546 Ki = 9000 nM T54156 CD9QO2 23645547 Ki = 1300 nM T54156 C25YLZ 23645548 Ki = 100 nM T54156 C4R2DA 23645953 Ki > 300000 nM T54156 CWN3I4 23645959 Ki > 300000 nM T54156 CL1KC0 23652834 IC50 = 7.83 nM T54156 COIZ43 23655713 IC50 = 821 nM T54156 CURM98 23655714 IC50 > 100000 nM T54156 CO90JC 23655717 IC50 = 1300 nM T54156 C3M2NQ 23655718 IC50 = 1350 nM T54156 C56NMQ 23655910 IC50 = 35000 nM T54156 C9QZX5 23655911 IC50 = 6930 nM T54156 CA8W3K 23656106 IC50 = 281 nM T54156 CU4R7T 23656291 IC50 = 50 nM T54156 CVZ2M1 23656293 IC50 = 69 nM T54156 CL5C1I 23656295 IC50 = 103 nM T54156 CZP12E 23656450 IC50 = 23 nM T54156 CA2PY5 23657418 IC50 = 614 nM T54156 CN9TY1 23657419 IC50 = 1330 nM T54156 C9FHZ1 23657421 IC50 = 51 nM T54156 CY9LF1 23657422 IC50 = 0.5 nM T54156 C28SPW 23657691 IC50 = 15000 nM T54156 CVJ1T7 23657695 IC50 = 10000 nM T54156 CAL05Q 23657697 IC50 = 9820 nM T54156 C6AW7U 23692637 IC50 > 100000 nM T54156 C7KF1N 23729138 IC50 = 120 nM T54156 C35QME 24742028 IC50 = 7 nM T54156 CY6KA0 24755074 IC50 = 67000 nM T54156 CQCJ17 24768595 IC50 = 0.46 nM T54156 CWLT01 24806172 IC50 = 7.8 nM T54156 CN59KZ 24806173 IC50 = 286 nM T54156 CH4X8K 24806175 IC50 = 0.52 nM T54156 C9RW0A 24806176 IC50 = 1.9 nM T54156 C18FRG 24807817 IC50 > 100000 nM T54156 CW3X0F 24852010 IC50 = 0.87 nM T54156 C2U0NS 24852011 IC50 = 5 nM T54156 C6YPS8 24852048 IC50 = 2.4 nM T54156 CUK6F1 24852487 IC50 = 31 nM T54156 C0MPV5 24852489 IC50 = 21.5 nM T54156 CNR3U7 24866945 IC50 > 100000 nM T54156 CRZ7Y6 24868315 IC50 = 19.6 nM T54156 C4UEM5 24871537 Ki > 50000 nM T54156 CP2L5B 24871655 Ki > 50000 nM T54156 CFL04M 24881245 IC50 = 200000 nM T54156 CLIC14 24881246 IC50 = 20000 nM T54156 C3U8ZQ 24882385 IC50 = 3050 nM T54156 C02WIB 24882535 IC50 = 5.5 nM T54156 C4FI5C 24901479 IC50 = 25703.96 nM T54156 C4SP3O 24936157 IC50 = 0.43 nM T54156 CBUA83 24936183 IC50 = 4 nM T54156 CQ2K9H 24936215 IC50 = 3048 nM T54156 C78OAU 24944977 IC50 = 830 nM T54156 CO6CJ5 24945161 IC50 = 3700 nM T54156 C1C0NX 24945244 IC50 = 18000 nM T54156 CLTQ28 24945246 IC50 = 1120 nM T54156 C7ZA6S 24945247 IC50 = 2500 nM T54156 CH3O0V 24951588 IC50 = 23 nM T54156 C8I4PT 24951589 IC50 = 2.8 nM T54156 C2Q1BK 24951590 IC50 = 1.3 nM T54156 COMJ45 24951950 IC50 = 20 nM T54156 C3JGU2 24951952 IC50 = 1.5 nM T54156 CC7U2T 24951953 IC50 = 0.54 nM T54156 CV86KA 24952316 IC50 = 0.62 nM T54156 CYJ2E9 24952318 IC50 = 472 nM T54156 CYKM71 24952674 IC50 = 14 nM T54156 C7MC8J 24952678 IC50 = 2.4 nM T54156 C0ZB8O 24953024 IC50 = 1.9 nM T54156 C5Z8XR 24953380 IC50 = 17 nM T54156 C2LN5E 24953381 IC50 = 256 nM T54156 CT2N3H 24953730 IC50 = 3.2 nM T54156 C1KH2Q 24953731 IC50 = 4.8 nM T54156 C0Q5BT 24954067 IC50 = 2.5 nM T54156 C6FI8O 24954068 IC50 = 1.1 nM T54156 CN29BR 24954070 IC50 = 2 nM T54156 CL1YO0 24954431 IC50 = 0.46 nM T54156 C3H9EO 24954432 IC50 = 2.3 nM T54156 CB60LR 24954795 IC50 = 8.8 nM T54156 C7P5YH 24954798 IC50 = 0.68 nM T54156 C5BG6I 24955154 IC50 = 91 nM T54156 CCE45B 24955155 IC50 = 47 nM T54156 CH53AG 24955156 IC50 = 44 nM T54156 CZC1P7 24955511 IC50 = 4.7 nM T54156 CL2G8J 24955513 IC50 = 68 nM T54156 CXG36M 24955514 IC50 = 1.7 nM T54156 CXO9Y4 24955857 IC50 = 3.8 nM T54156 CKY2F6 24955858 IC50 = 2.9 nM T54156 C4LJ8N 24955859 IC50 = 5.4 nM T54156 CX4MY3 24955861 IC50 = 12 nM T54156 CR29SO 24956227 IC50 = 124 nM T54156 CSM26P 24956228 IC50 = 13 nM T54156 C13JHO 24956229 IC50 = 0.52 nM T54156 C01QMC 24956580 IC50 = 243 nM T54156 C8M5PJ 24956581 IC50 = 28 nM T54156 CC90AR 24956582 IC50 = 344 nM T54156 CQH6I4 24956585 IC50 = 31 nM T54156 CHJ50Q 24956943 IC50 = 7.1 nM T54156 CN2AS5 24956945 IC50 = 121 nM T54156 C2HN8M 24956948 IC50 = 1.8 nM T54156 C2VEZ0 24957161 IC50 = 295 nM T54156 CNCA57 25004194 Ki = 4.677 nM T54156 CAQ9Z1 25022681 Ki > 2128 nM T54156 CVR52U 25066764 IC50 = 1300 nM T54156 CD2KA4 25102047 IC50 = 9 nM T54156 CRW96X 25102048 IC50 = 8.6 nM T54156 CQ3O9P 25102050 IC50 = 6.5 nM T54156 CSHA26 25102051 IC50 = 6.4 nM T54156 C7ADO2 25102197 IC50 = 2.9 nM T54156 C1TNQ3 25141117 IC50 = 3 nM T54156 CR35QP 25144971 IC50 > 10000 nM T54156 C0Y5BC 25145683 IC50 > 2500 nM T54156 CB7V8Y 25147773 IC50 = 0.21 nM T54156 C3KF1V 25178145 IC50 = 0.51 nM T54156 C8PMK7 25178356 IC50 > 300000 nM T54156 CG5Y2R 25178357 IC50 = 27.7 nM T54156 C4PZY6 25180866 IC50 = 62 nM T54156 CEP9Q2 25180867 IC50 = 0.77 nM T54156 C7U1YC 25181080 IC50 = 53.7 nM T54156 C85HLG 25181081 IC50 = 66 nM T54156 CHR2P1 25183768 Ki > 25000 nM T54156 CZ8CR1 25190501 Ki > 2128 nM T54156 CO8CD1 25190502 Ki > 2128 nM T54156 C0R6MU 25212135 IC50 = 37360 nM T54156 C9GCO4 28602444 IC50 > 150000 nM T54156 CPO1Z3 44123600 IC50 = 10 nM T54156 CWS64Q 44143474 IC50 > 12000 nM T54156 C06IJY 44143476 IC50 = 12000 nM T54156 CH1IR0 44144307 IC50 = 10170 nM T54156 CT80ED 44219901 IC50 = 1100 nM T54156 C94JVY 44219902 IC50 = 2300 nM T54156 C7J6GH 44219903 IC50 = 110 nM T54156 C9J7WL 44219904 IC50 = 4400 nM T54156 CRQ71E 44219905 IC50 = 3200 nM T54156 C4Z0ID 44219906 IC50 = 680 nM T54156 CRNA25 44220092 IC50 = 250 nM T54156 C9T5ZF 44220093 IC50 = 69 nM T54156 CV38TE 44222825 IC50 = 44 nM T54156 CJI73R 44222826 IC50 = 77 nM T54156 CGQ30N 44222827 IC50 = 160 nM T54156 CCI64J 44224245 IC50 = 318 nM T54156 CLRT69 44247751 IC50 = 0.8 nM T54156 C7U4XP 44250718 IC50 = 12490 nM T54156 CAR34Y 44263877 IC50 = 24.1 nM T54156 CEV08N 44263913 IC50 = 1.8 nM T54156 C5ZI0X 44263926 IC50 = 1 nM T54156 CO3C1E 44263994 IC50 = 5.5 nM T54156 C9XJ7U 44264020 IC50 = 52.5 nM T54156 C6L0MJ 44264021 IC50 = 4.1 nM T54156 CJ1WE7 44264036 IC50 = 3.3 nM T54156 C50QFR 44264375 IC50 = 4.2 nM T54156 CDL25C 44265349 Ki = 2.8 nM T54156 C3W4QO 44265401 Ki = 87 nM T54156 C2Q3JV 44265407 Ki = 3422 nM T54156 CN59QT 44265437 Ki > 2000 nM T54156 CZA61K 44265475 Ki = 347 nM T54156 CD4A7F 44265476 Ki = 277 nM T54156 CT6FK0 44265480 Ki = 4.2 nM T54156 C67HUL 44265485 Ki = 5.4 nM T54156 CH0O3I 44265492 Ki = 1085 nM T54156 C0DFG7 44265501 Ki = 150 nM T54156 CCM8K0 44265512 Ki = 17.2 nM T54156 CB3E6O 44265527 Ki < 2.11 nM T54156 C3YK0O 44268937 IC50 = 1000 nM T54156 C5DG8Z 44268941 IC50 = 200 nM T54156 C3SGT4 44268967 IC50 = 900 nM T54156 C1Z0GQ 44269012 IC50 = 1000 nM T54156 C18VGL 44269017 IC50 = 10000 nM T54156 C8S2FJ 44270678 IC50 = 6 nM T54156 C2BUH0 44270679 IC50 = 5 nM T54156 C4OJK9 44270703 IC50 = 4 nM T54156 C8MUJ3 44270704 IC50 = 780 nM T54156 C0K3RP 44270736 IC50 = 1.4 nM T54156 CLMO84 44270737 IC50 = 19 nM T54156 CKL2C3 44270739 IC50 = 30 nM T54156 C4B0LP 44270775 IC50 = 640 nM T54156 C1WTN7 44270802 IC50 = 1.4 nM T54156 CVG61X 44270805 IC50 = 4500 nM T54156 CNU41R 44270901 IC50 = 20 nM T54156 CDX36Y 44270985 IC50 = 24 nM T54156 CFR81A 44271005 IC50 = 12 nM T54156 CRF2Z5 44271421 IC50 = 7.14 nM T54156 CG92WS 44272353 IC50 = 166 nM T54156 CO2Z6K 44272475 IC50 = 2 nM T54156 C63KSL 44272540 IC50 = 28 nM T54156 CG7X5F 44272675 IC50 = 14 nM T54156 CEHR24 44272853 IC50 = 45 nM T54156 CJ3MV2 44274642 Ki > 2128 nM T54156 CC2QR7 44281720 Ki = 13 nM T54156 CN23FC 44282968 IC50 = 2500 nM T54156 C2TV5I 44282969 IC50 = 150 nM T54156 CG3LF0 44282970 IC50 = 150 nM T54156 C6S3GN 44283598 IC50 = 5 nM T54156 CXE73H 44283613 IC50 = 7 nM T54156 CP3L2U 44283938 IC50 = 595 nM T54156 C3UB9V 44286654 Ki = 118.37 nM T54156 CB07MX 44286663 Ki = 98.2 nM T54156 C3KXY9 44286674 Ki = 12 nM T54156 CJ7VW3 44291166 IC50 = 2.5 nM T54156 C75IEN 44291420 IC50 = 0.2 nM T54156 CF21CS 44291532 IC50 = 0.2 nM T54156 CU75TB 44291559 IC50 = 7 nM T54156 C06JAO 44291626 IC50 = 8 nM T54156 C4LI6F 44293416 Ki = 0.13 nM T54156 C5XS0I 44294322 Ki = 404 nM T54156 CAFB18 44296974 Ki = 1839 nM T54156 C8NTY1 44299442 IC50 = 80 nM T54156 CE34KO 44299443 IC50 = 84 nM T54156 C7Z0IF 44299460 IC50 = 82 nM T54156 C06NTZ 44299503 IC50 = 49 nM T54156 CQSA71 44299538 IC50 = 41 nM T54156 C2LXS8 44299719 IC50 = 71 nM T54156 C03HUT 44299735 IC50 = 24 nM T54156 C6HY7N 44299870 IC50 = 41 nM T54156 COV3W7 44299871 IC50 = 38 nM T54156 C9R2FL 44299872 IC50 = 34 nM T54156 CTGR41 44299873 IC50 = 21 nM T54156 C8K6VC 44299880 IC50 = 19 nM T54156 C2WZ7S 44299893 IC50 = 15 nM T54156 CG3EJ5 44299894 IC50 = 11 nM T54156 CD5Y6C 44299895 IC50 > 1000 nM T54156 CRDX61 44299910 IC50 = 71 nM T54156 C79UQM 44299911 IC50 = 42 nM T54156 C6PDF1 44299928 IC50 = 102 nM T54156 C5RSX9 44300181 IC50 = 24000 nM T54156 C2FSR6 44302165 IC50 = 1.5 nM T54156 CALD50 44304020 Ki > 2000 nM T54156 C0IJ9D 44304112 Ki = 23.7 nM T54156 CSVK45 44304230 Ki > 2000 nM T54156 C5QUK2 44308295 Ki = 98 nM T54156 C2E4IT 44308297 Ki = 17 nM T54156 C0K4UQ 44308298 Ki = 29 nM T54156 CCRW50 44308304 Ki = 17 nM T54156 CZF5S2 44308327 Ki = 89 nM T54156 COE56H 44308377 Ki = 21 nM T54156 C7OT6S 44308488 Ki = 33 nM T54156 CI2Z0H 44308525 Ki = 28 nM T54156 CU0J5A 44308623 Ki = 73 nM T54156 CSEB94 44308624 Ki = 24 nM T54156 CST39W 44308640 Ki = 34 nM T54156 C5AM6P 44308844 IC50 = 1642.27 nM T54156 C4SJF3 44309329 IC50 = 2 nM T54156 C7ED1H 44309330 IC50 = 1 nM T54156 C1E3KF 44309437 IC50 = 3 nM T54156 CH3SU2 44309482 IC50 = 3448 nM T54156 C6N5SL 44309531 IC50 = 152 nM T54156 CO7TS8 44309532 IC50 = 153 nM T54156 CQ7Z0W 44309533 IC50 = 189 nM T54156 CJ0L4P 44309550 IC50 = 8 nM T54156 CKEU31 44309629 IC50 = 2365 nM T54156 C6J3WN 44309662 IC50 = 7 nM T54156 CY96UH 44309686 IC50 = 4 nM T54156 C49MHR 44309863 IC50 = 952 nM T54156 CMW0U4 44309879 IC50 = 2 nM T54156 CK6BT0 44309901 IC50 = 232 nM T54156 C5WZR7 44309939 IC50 = 125 nM T54156 CZUY51 44310789 Ki = 1.7 nM T54156 CH92OI 44310813 Ki = 3.5 nM T54156 CI4Y5N 44310825 Ki = 6.9 nM T54156 C5W8QH 44310847 Ki = 1.7 nM T54156 CLQV12 44310863 Ki = 0.83 nM T54156 CR70EA 44310887 Ki = 1.6 nM T54156 CJ9T1F 44310904 Ki = 1.5 nM T54156 CN9P5A 44310921 Ki = 1.3 nM T54156 CXB76U 44310932 Ki = 0.99 nM T54156 CMW5G3 44310933 Ki = 6.5 nM T54156 CBY0T1 44310973 Ki = 6.3 nM T54156 C5D9FS 44311011 Ki = 0.58 nM T54156 C95RKF 44311052 Ki = 3 nM T54156 C2GC9W 44311172 Ki = 5.3 nM T54156 C0K1IL 44311187 Ki = 1.5 nM T54156 CL3CS0 44311254 Ki = 26 nM T54156 CV63JP 44311265 Ki = 2.5 nM T54156 CS56ER 44311267 Ki = 74 nM T54156 C5MBT7 44311268 Ki = 3.8 nM T54156 CM64HK 44311313 Ki = 1.7 nM T54156 CU5X4G 44311331 Ki = 2.7 nM T54156 CLQ48B 44311332 Ki = 3.6 nM T54156 C5AO7Z 44311335 Ki = 0.96 nM T54156 C78TEU 44311349 Ki = 2.8 nM T54156 CJEM64 44311491 Ki = 2.5 nM T54156 C2W5NQ 44311510 Ki = 2.3 nM T54156 C2MIT8 44311525 Ki = 0.7 nM T54156 CP7L6Q 44311566 Ki = 4.1 nM T54156 C0B4HZ 44312333 Ki = 23.99 nM T54156 CJ9OE7 44313735 IC50 = 2.4 nM T54156 C5HAY4 44313736 IC50 = 4.3 nM T54156 CKLJ71 44313754 IC50 = 2.8 nM T54156 CX4BM9 44313996 IC50 = 237 nM T54156 CK9XB7 44314087 IC50 = 1.1 nM T54156 C8MRB1 44314322 IC50 = 0.092 nM T54156 CB6UL7 44314349 IC50 = 5.5 nM T54156 C3R0DL 44314366 IC50 = 1.1 nM T54156 C92MGV 44314566 IC50 = 0.34 nM T54156 CLT6E0 44314618 IC50 = 120 nM T54156 CSY78M 44315028 Ki = 290 nM T54156 CDZ5O3 44315029 Ki = 1500 nM T54156 COA01P 44315179 Ki = 19200 nM T54156 CL32FZ 44315221 Ki = 620 nM T54156 CDN4Y5 44315222 Ki = 184 nM T54156 CKAL69 44315860 IC50 = 4 nM T54156 C0HR5Q 44316157 IC50 = 6 nM T54156 C5RJ6F 44316310 IC50 = 4 nM T54156 CSA5P7 44316333 IC50 = 1.995 nM T54156 CS5V0J 44316334 IC50 = 64 nM T54156 CS7D5E 44317086 IC50 = 14 nM T54156 CH70XB 44317451 IC50 = 181 nM T54156 C89IQW 44318090 IC50 = 18.7 nM T54156 CJU31O 44321285 Ki = 6 nM T54156 C41VFA 44321286 Ki = 10 nM T54156 C5S2ZU 44321484 Ki = 55 nM T54156 CLQ23M 44321485 Ki = 65 nM T54156 CHF76Q 44321540 Ki = 6 nM T54156 CVOL49 44321593 Ki = 44 nM T54156 CB97GK 44321601 Ki = 35 nM T54156 CT0O7Y 44321602 Ki = 245 nM T54156 CU62BP 44321746 Ki = 10 nM T54156 CQU2K9 44321782 Ki = 110 nM T54156 CV8T3N 44321783 Ki = 13 nM T54156 CIBO50 44321801 Ki = 3 nM T54156 C4E8GU 44321802 Ki = 55 nM T54156 CYDN18 44321803 Ki = 22 nM T54156 C7Z4DQ 44321887 Ki = 7 nM T54156 CFJ20T 44321932 Ki = 8 nM T54156 C2E3RF 44321966 Ki = 30 nM T54156 CW9S1N 44321967 Ki = 675 nM T54156 C1FI3O 44321975 Ki = 6 nM T54156 CLB8J6 44321976 Ki = 60 nM T54156 CR0KN1 44322209 Ki = 280 nM T54156 C5LE1P 44322210 Ki = 23 nM T54156 CQ7AW8 44322211 Ki = 44 nM T54156 CJY2O7 44322214 Ki = 110 nM T54156 CR9GI0 44322215 Ki = 70 nM T54156 C15WQO 44323336 IC50 = 2 nM T54156 C9UOW2 44323407 IC50 = 31 nM T54156 C4C1WD 44323426 IC50 = 3.3 nM T54156 C85JGD 44323430 IC50 = 157 nM T54156 CKP12T 44323431 IC50 = 9.2 nM T54156 C4R8OD 44323432 IC50 = 18 nM T54156 COQ6U7 44323456 IC50 = 60 nM T54156 CL07GT 44323526 IC50 = 9.1 nM T54156 CZRF63 44323527 IC50 = 23 nM T54156 CT9M4F 44323539 IC50 = 4.8 nM T54156 CQG24X 44323540 IC50 = 4 nM T54156 CO0S9J 44325072 Ki = 0.93 nM T54156 C4R9LM 44325085 Ki = 6.1 nM T54156 CL8MD0 44325156 Ki = 64 nM T54156 CV3S9G 44325157 Ki = 82 nM T54156 C9MD1A 44325159 Ki = 780 nM T54156 C6R4NI 44325225 Ki = 310 nM T54156 C3M2XY 44325277 Ki = 157 nM T54156 CA4FQ5 44325443 Ki = 47 nM T54156 C7V5EF 44326167 IC50 = 40 nM T54156 C93HSL 44326184 IC50 = 30 nM T54156 CY3I9B 44326185 IC50 = 5 nM T54156 C23OQF 44326225 IC50 = 30 nM T54156 CY3GH5 44326232 IC50 = 32 nM T54156 C6E9IV 44326443 IC50 = 50 nM T54156 C2ZH0F 44327181 IC50 = 794.33 nM T54156 C8V3AO 44327386 IC50 = 224 nM T54156 C0UC5H 44327407 IC50 = 41.69 nM T54156 C6TPB1 44327409 IC50 = 128.82 nM T54156 C8ZI0P 44327432 IC50 = 346.74 nM T54156 CVJ9Q6 44327443 IC50 = 67.61 nM T54156 C4R9WM 44327681 IC50 = 10.96 nM T54156 CR40TV 44327695 IC50 = 74 nM T54156 C6IM7G 44327755 IC50 = 158.49 nM T54156 C85QTP 44328155 IC50 = 500 nM T54156 CZQ6N7 44328189 IC50 > 100000 nM T54156 CHU2P7 44328876 IC50 = 2 nM T54156 C0KA4S 44328937 IC50 = 4 nM T54156 CLT8B6 44328971 IC50 = 2 nM T54156 C7J0ZI 44329016 IC50 = 2 nM T54156 CMLA39 44329018 IC50 = 17 nM T54156 CW24VN 44329040 IC50 = 2 nM T54156 C9J0VO 44329253 IC50 = 2 nM T54156 C3YAF6 44329898 IC50 = 28000 nM T54156 C9R1ZE 44330132 IC50 = 31000 nM T54156 CLU8I7 44330135 IC50 = 40000 nM T54156 C1IE0S 44330147 IC50 > 100000 nM T54156 CPG7N2 44330149 IC50 = 53000 nM T54156 CYP6S4 44330152 IC50 = 12000 nM T54156 CMGA28 44330163 IC50 = 50000 nM T54156 CD0L6S 44331932 IC50 = 3 nM T54156 CHIG68 44331976 IC50 = 10 nM T54156 CF4JN0 44331983 IC50 = 2 nM T54156 CG2AH4 44331984 IC50 = 2 nM T54156 CPB96A 44332003 IC50 = 5 nM T54156 C6RE3I 44332107 IC50 = 0.5 nM T54156 C3L1HQ 44332161 IC50 = 7 nM T54156 CG2Q8W 44332306 IC50 = 199 nM T54156 CY0MQ9 44332313 IC50 = 14 nM T54156 C5NG0R 44334948 IC50 = 0.2 nM T54156 CFP3X8 44334949 IC50 = 7 nM T54156 CV5RF0 44334963 IC50 = 138 nM T54156 C4AOZ7 44334981 IC50 = 50 nM T54156 CXW59C 44334982 IC50 = 4.4 nM T54156 CCH1W8 44334983 IC50 = 0.9 nM T54156 CQ0UI1 44335017 IC50 = 9.2 nM T54156 CX58SB 44335240 IC50 = 0.9 nM T54156 CA96JG 44335285 IC50 = 2.8 nM T54156 CM3F2G 44337397 IC50 = 850 nM T54156 C9L3HU 44337570 IC50 = 190 nM T54156 CL9I4M 44341538 Ki = 4200 nM T54156 CE3MT4 44341611 Ki = 3910 nM T54156 CJTZ45 44341652 Ki = 148000 nM T54156 C2SZB1 44342614 IC50 = 3 nM T54156 C8G7WL 44344564 Ki = 330 nM T54156 CD43AB 44344565 Ki = 20 nM T54156 CTQ6P4 44344631 IC50 = 30400 nM T54156 CBH9I5 44344658 IC50 = 560 nM T54156 CC29QO 44344739 Ki = 5600 nM T54156 CWA42F 44344746 Ki = 11 nM T54156 CQPN17 44344749 Ki = 1.3 nM T54156 CL41FG 44344753 Ki = 500 nM T54156 CCF94Z 44349787 IC50 = 3.3 nM T54156 C1L2GF 44350073 IC50 = 62 nM T54156 CQ5RN6 44350101 IC50 = 642 nM T54156 CE2X3Q 44350116 IC50 > 100 nM T54156 CO9R4W 44356376 Ki > 2128 nM T54156 C3MZA1 44356386 Ki > 2128 nM T54156 CH1E2S 44356406 Ki > 2128 nM T54156 C84LUM 44356631 Ki > 2128 nM T54156 CG6T9A 44356632 Ki > 2128 nM T54156 C3WFH7 44356634 Ki > 2128 nM T54156 CB8KY4 44356635 Ki > 2128 nM T54156 COIA82 44356636 Ki > 2128 nM T54156 C4BU6T 44356644 Ki > 2128 nM T54156 CH9YT4 44356659 Ki > 2128 nM T54156 C68LMR 44356675 Ki > 2128 nM T54156 C69YIP 44356686 Ki > 2128 nM T54156 CT05XN 44356687 Ki 876 nM T54156 CML03W 44356689 Ki > 2128 nM T54156 CQ4NP5 44356690 Ki > 2128 nM T54156 CE8U2Y 44356714 Ki > 2128 nM T54156 CCY5U3 44356804 Ki = 450 nM T54156 C27LMU 44356852 Ki > 2128 nM T54156 CTU64D 44356889 Ki > 2128 nM T54156 C4TM1I 44356890 Ki > 2128 nM T54156 C1WA4B 44356906 Ki > 2128 nM T54156 C50ELY 44356907 Ki > 2128 nM T54156 CVU8L2 44356924 Ki > 2128 nM T54156 CD1GW2 44356953 Ki > 465 nM T54156 CR41QN 44356969 Ki > 1656 nM T54156 C3BT0N 44356971 Ki = 209 nM T54156 C81OIZ 44356983 Ki > 2128 nM T54156 CHNC03 44356993 Ki > 2128 nM T54156 C9Z3RT 44356998 Ki > 2128 nM T54156 CR4A7G 44356999 Ki = 296 nM T54156 C2VS6P 44357000 Ki = 768 nM T54156 CES1G8 44357007 Ki > 2128 nM T54156 C6NQ7K 44357012 Ki = 306 nM T54156 C2HIN3 44357023 Ki > 2128 nM T54156 CI4JO7 44357024 Ki 1358 nM T54156 CW4VQ3 44357029 Ki > 2128 nM T54156 C2AIT6 44357209 Ki > 2128 nM T54156 CJK2P7 44357220 Ki > 2128 nM T54156 CIX6G5 44357225 Ki > 2128 nM T54156 C3IW9L 44360784 IC50 = 0.5 nM T54156 CGQ92A 44364037 IC50 = 130 nM T54156 C36YLM 44364111 IC50 = 248 nM T54156 CN4T7Q 44364119 IC50 = 0.25 nM T54156 CH4TE7 44364121 IC50 = 35 nM T54156 CPE91Y 44364122 IC50 = 40 nM T54156 CG2X0C 44364224 IC50 = 335 nM T54156 C1F8XN 44364249 IC50 = 46 nM T54156 CWM47H 44364250 IC50 = 100 nM T54156 C0W5TL 44364251 IC50 = 3118 nM T54156 C3TPO7 44364266 IC50 = 1882 nM T54156 CJ2B8F 44364280 IC50 = 4100 nM T54156 C92OKS 44369679 Ki = 14.2 nM T54156 C63WRQ 44369680 Ki > 800 nM T54156 CHV7Z8 44369681 Ki = 5.53 nM T54156 CX4ZU6 44369702 Ki > 800 nM T54156 C8ZK2I 44369876 Ki = 24.1 nM T54156 CDCT62 44372514 IC50 = 730 nM T54156 CQ5UR4 44372530 IC50 = 800 nM T54156 CL98HN 44372668 IC50 > 1000000 nM T54156 C1QWA3 44374051 IC50 = 14 nM T54156 CX01WF 44374220 IC50 = 70 nM T54156 C40TSF 44374235 IC50 = 76 nM T54156 C1I6QU 44374342 IC50 = 580 nM T54156 CZYL14 44374353 IC50 = 12 nM T54156 CGK04Y 44374370 IC50 = 63 nM T54156 C4M3CU 44380421 Ki < 1 nM T54156 C0CH2Q 44380422 Ki < 1 nM T54156 CBLY46 44380446 Ki = 2 nM T54156 C0F6ZP 44380458 Ki = 5 nM T54156 C1VY9Q 44380628 Ki = 1 nM T54156 C4H8SW 44380647 Ki = 34 nM T54156 CY03NT 44380706 Ki = 5 nM T54156 CJ5W2S 44381004 Ki = 149 nM T54156 C82UHB 44381005 Ki = 1 nM T54156 C8A9FK 44381033 Ki < 1 nM T54156 C3LIF2 44381197 Ki = 4 nM T54156 C27DGC 44381207 Ki = 2 nM T54156 C70VDN 44381208 Ki = 2 nM T54156 CYE90S 44383704 Ki = 16.7 nM T54156 C4O9DP 44383747 Ki = 0.08 nM T54156 C0W2SV 44383786 Ki = 0.1 nM T54156 C2UNW6 44383789 Ki = 2.03 nM T54156 CV0T6G 44383797 Ki = 250 nM T54156 C6V9FQ 44383801 Ki = 5.22 nM T54156 CV8UX5 44383829 Ki = 0.6 nM T54156 C9NIT7 44383842 Ki = 350 nM T54156 C2SZ1O 44383843 Ki = 3300 nM T54156 CCY30B 44383847 Ki = 6.47 nM T54156 C7MLD8 44383849 Ki = 4.56 nM T54156 C4Y0PX 44383857 Ki = 600 nM T54156 C13LRY 44383990 Ki = 3300 nM T54156 C9F5LS 44384003 Ki = 59.2 nM T54156 CSM3P7 44384004 Ki = 95.6 nM T54156 CO9LJ6 44384005 Ki = 278 nM T54156 CDQV80 44384020 Ki = 150 nM T54156 CA2L3U 44384021 Ki = 4400 nM T54156 CT1MN8 44384090 Ki = 9000 nM T54156 CB16LN 44384094 Ki = 8200 nM T54156 C8OKQ9 44384146 Ki = 4000 nM T54156 CJ4NV9 44384173 Ki = 32.1 nM T54156 C5C3LY 44384231 Ki = 800 nM T54156 CILQ34 44384272 Ki = 14000 nM T54156 CIJ61R 44384273 Ki = 900 nM T54156 C7B3AN 44384343 Ki = 11 nM T54156 CQ2UE9 44384356 Ki = 2000 nM T54156 C4B9NU 44384357 Ki = 80.1 nM T54156 CL59ZH 44384393 Ki = 7500 nM T54156 CC81JP 44384395 Ki = 1.13 nM T54156 C14RMP 44384416 Ki = 500 nM T54156 CKG95Y 44384455 Ki = 316 nM T54156 C5MO9Q 44384474 Ki = 3200 nM T54156 C96PAY 44384542 Ki = 3.42 nM T54156 C7HA0F 44384590 Ki = 51.9 nM T54156 C5ZYN1 44384591 Ki = 41.8 nM T54156 CVZ42A 44384592 Ki = 88.8 nM T54156 C49TAV 44384649 Ki = 42.7 nM T54156 CALI01 44384650 Ki = 6.36 nM T54156 C8SCB5 44384659 Ki > 800 nM T54156 C7A2HC 44384755 Ki = 5.2 nM T54156 CL51XE 44384756 Ki = 3.8 nM T54156 CD2PM4 44384761 Ki = 0.31 nM T54156 CJH8P4 44384762 Ki = 14.2 nM T54156 C0RXF4 44384804 Ki = 1000 nM T54156 CH3M5X 44384813 Ki = 23.2 nM T54156 C59NBH 44384814 Ki = 6.57 nM T54156 C3EV2A 44384940 IC50 = 164 nM T54156 C0XE8K 44384941 IC50 = 12000 nM T54156 C5AE0O 44384972 Ki = 38.3 nM T54156 CUMQ67 44384980 Ki = 600 nM T54156 C3IJO9 44384994 IC50 > 50000 nM T54156 C3CG5I 44385039 Ki = 3000 nM T54156 CE7V9A 44385250 Ki = 44000 nM T54156 CE5RJ0 44385333 Ki = 5500 nM T54156 C2FKP7 44385334 Ki = 800 nM T54156 CHT2D6 44385339 Ki = 100 nM T54156 CK7RP9 44385344 Ki = 9.12 nM T54156 CZ6PU7 44389401 Ki = 1.9 nM T54156 CO4W0Y 44389552 Ki = 0.7 nM T54156 CWQ19I 44389560 IC50 = 13 nM T54156 C5R4EW 44389591 IC50 = 4517 nM T54156 C89FTQ 44393434 Ki > 5000 nM T54156 CCO3S9 44393444 Ki > 2100 nM T54156 CNO4P6 44393516 Ki > 2100 nM T54156 C5OIK4 44393520 Ki > 2100 nM T54156 C80NZE 44394179 Ki > 2100 nM T54156 C1TWP6 44394594 Ki > 100000 nM T54156 CG01SR 44394595 Ki > 100000 nM T54156 CV6YR1 44394601 Ki = 22000 nM T54156 CG6YH0 44394631 Ki = 32000 nM T54156 C6OM9B 44394637 Ki = 94000 nM T54156 CXD05N 44394645 Ki > 100000 nM T54156 CZ05UP 44394668 Ki = 88000 nM T54156 CAFL18 44394671 Ki = 94000 nM T54156 CGQ98X 44394681 Ki = 8000 nM T54156 CQM90E 44394682 Ki = 65000 nM T54156 C28HVB 44394702 Ki > 200000 nM T54156 C8MY4S 44394703 Ki > 100000 nM T54156 CY3B2Q 44394721 Ki > 2000000 nM T54156 C12XGC 44394727 Ki > 2000000 nM T54156 CGS56H 44394744 Ki > 100000 nM T54156 CK5X6F 44394758 Ki = 81000 nM T54156 C6WA3L 44394765 Ki > 100000 nM T54156 CUK01T 44394796 Ki > 100000 nM T54156 CCEI41 44394814 Ki > 4000000 nM T54156 C79OYF 44394821 Ki = 33000 nM T54156 C5BSH2 44394838 Ki = 24000 nM T54156 CVX1H4 44394873 Ki = 40000 nM T54156 C8Y4FP 44394879 Ki = 68000 nM T54156 CZB81D 44395506 IC50 = 11 nM T54156 C4L1FI 44398813 Ki = 41.78 nM T54156 CGJF83 44398848 Ki = 3.42 nM T54156 CNC7H6 44398880 Ki = 42.66 nM T54156 CV9I8C 44398899 Ki = 38.28 nM T54156 C02KPY 44398985 Ki = 6.353 nM T54156 CB8I6O 44398986 Ki = 0.1 nM T54156 CQI8A9 44399042 Ki = 5.047 nM T54156 C9SKI1 44399043 Ki = 4.56 nM T54156 CLPU49 44399044 Ki = 0.07943 nM T54156 C6PK9T 44399060 Ki = 277.97 nM T54156 CEK4I7 44399074 Ki = 349 nM T54156 CBM9J4 44399087 Ki = 59.16 nM T54156 CNI8V0 44399101 Ki = 1.13 nM T54156 C2WVS4 44399108 Ki = 16.71 nM T54156 CR89OC 44399124 Ki = 6.577 nM T54156 CB26HI 44399144 Ki = 0.3097 nM T54156 CC7S9Y 44399156 Ki = 32.14 nM T54156 C9F4OH 44399188 Ki = 95.5 nM T54156 C4M9FA 44399208 Ki = 6.471 nM T54156 CW6F7Z 44399219 Ki = 2.028 nM T54156 CRWF05 44399220 Ki = 0.5998 nM T54156 CJN52A 44399235 Ki = 14.19 nM T54156 CYUM48 44399258 Ki = 80.17 nM T54156 CHL9S2 44399294 Ki = 850 nM T54156 CD49UI 44399312 Ki > 2130 nM T54156 CIA8T3 44399555 Ki > 2130 nM T54156 C8PR7S 44400182 IC50 = 4 nM T54156 CQ9F0K 44400232 IC50 = 6 nM T54156 C91POV 44402021 IC50 = 983 nM T54156 CYCJ78 44402280 IC50 = 8.3 nM T54156 CWG3M4 44402281 IC50 > 30000 nM T54156 C7Z0OH 44404761 IC50 = 209 nM T54156 CHM26J 44406652 Ki = 6600 nM T54156 C6YG5S 44406678 IC50 = 2.7 nM T54156 CB5ZS0 44411587 IC50 = 114 nM T54156 C4Z0BX 44411591 IC50 > 10000 nM T54156 CHV64P 44411592 IC50 = 4.4 nM T54156 CL6IG9 44411599 IC50 = 120 nM T54156 C6IKL1 44411602 IC50 = 0.5 nM T54156 CM2UL0 44411603 IC50 = 1.4 nM T54156 CBT4E7 44411614 IC50 = 25 nM T54156 CH8B4W 44411639 IC50 = 9.7 nM T54156 CS74LI 44411640 IC50 = 101 nM T54156 C43HTC 44411693 IC50 = 15 nM T54156 C8HSN2 44411697 IC50 = 4.9 nM T54156 CKQ8P6 44411698 IC50 = 0.96 nM T54156 CVQ82B 44411701 IC50 = 31 nM T54156 C87VNZ 44411702 IC50 = 0.8 nM T54156 C83MTG 44411776 IC50 = 1.6 nM T54156 CT1A8Q 44411815 IC50 > 10000 nM T54156 CQLV08 44411816 IC50 = 1049 nM T54156 CP16XL 44411819 IC50 = 14 nM T54156 C9COT4 44411820 IC50 = 53 nM T54156 C3Q8PM 44411822 IC50 = 20 nM T54156 CEB0S4 44411823 IC50 = 1.8 nM T54156 CRB85W 44411826 IC50 = 22 nM T54156 CV1NO8 44411829 IC50 = 5.1 nM T54156 CPH6V5 44411830 IC50 = 1.4 nM T54156 CRKL06 44411835 IC50 = 2124 nM T54156 C0FDM1 44411836 IC50 = 96.5 nM T54156 CUV27I 44411839 IC50 = 23 nM T54156 CD5KV9 44411846 IC50 = 258 nM T54156 C7CU1F 44411852 IC50 = 0.6 nM T54156 CA9OS4 44411865 IC50 = 1.2 nM T54156 C4X0GA 44413977 IC50 = 68 nM T54156 CQ8HK9 44413979 IC50 = 1070 nM T54156 CBT0P2 44413982 IC50 = 191 nM T54156 C9BA0V 44413987 IC50 = 907 nM T54156 CDUI73 44413992 IC50 = 19 nM T54156 CH2X6W 44413997 IC50 = 19 nM T54156 C2OJ4B 44414029 IC50 = 2120 nM T54156 CGDY32 44415219 IC50 = 29600 nM T54156 CZ5KM8 44421257 IC50 > 10000 nM T54156 CT5PC9 44422672 IC50 = 4.1 nM T54156 CS9D5U 44422720 IC50 = 0.56 nM T54156 CNWM05 44422723 IC50 = 24 nM T54156 C58LAY 44422724 IC50 = 59 nM T54156 CDQU41 44422736 IC50 = 170 nM T54156 CVUB56 44422737 IC50 = 160 nM T54156 CB8G2W 44422743 IC50 = 64 nM T54156 CFX42T 44422744 IC50 = 7100 nM T54156 C9EL7F 44422749 IC50 = 680 nM T54156 CY49HT 44423674 IC50 = 2200 nM T54156 CHI5G1 44423675 IC50 = 870 nM T54156 CFC3M6 44423676 IC50 = 330 nM T54156 CO24JF 44423677 IC50 = 3400 nM T54156 C7F9DB 44423678 IC50 = 33000 nM T54156 CJ6GW5 44423679 IC50 = 2000 nM T54156 CUKM29 44423680 IC50 = 1830 nM T54156 C3R0FS 44423681 IC50 = 370 nM T54156 C14DBJ 44423682 IC50 = 286 nM T54156 CK5H7O 44429877 IC50 = 90000 nM T54156 C8BHL5 44431844 IC50 > 2000 nM T54156 CR1DN9 44431845 IC50 > 2000 nM T54156 CHFB16 44431846 IC50 > 2000 nM T54156 C0C3ZT 44431847 IC50 > 2000 nM T54156 CS49GV 44431848 IC50 > 2000 nM T54156 C4AVK5 44431849 IC50 > 2000 nM T54156 C5DH4Q 44431850 IC50 > 2000 nM T54156 CLHE45 44431851 IC50 > 2000 nM T54156 CYG29L 44431852 IC50 > 2000 nM T54156 C4OF5L 44431853 IC50 > 2000 nM T54156 CWU7G8 44434565 IC50 > 100000 nM T54156 CF9HU5 44434566 IC50 = 45 nM T54156 CV3M6F 44434578 IC50 = 38 nM T54156 C70MGQ 44440455 Ki > 2128 nM T54156 CDY53F 44440460 Ki > 2128 nM T54156 CTB9P6 44440461 Ki = 179 nM T54156 C63RLK 44440462 Ki > 2128 nM T54156 C23JBO 44440463 Ki > 2128 nM T54156 CT9P3Y 44440464 Ki > 2128 nM T54156 CX32AM 44440465 Ki > 2128 nM T54156 C6FOC7 44440466 Ki > 2128 nM T54156 CMPX37 44440467 Ki > 2128 nM T54156 CV4F6Z 44440468 Ki > 2128 nM T54156 C6K8VB 44440469 Ki > 2128 nM T54156 C4Y0UM 44440470 Ki > 2128 nM T54156 CHU49A 44440471 Ki > 2128 nM T54156 C0HX1L 44445199 IC50 = 67000 nM T54156 CPQT35 44445200 IC50 = 62000 nM T54156 C2X6IP 44445201 IC50 = 69000 nM T54156 CSRB79 44445202 IC50 = 68000 nM T54156 C2O6KZ 44445203 IC50 = 94000 nM T54156 CASF34 44445204 IC50 = 69000 nM T54156 CQZ6M0 44445205 IC50 = 81000 nM T54156 CH7Z5M 44445206 IC50 = 68000 nM T54156 C71CPO 44445207 IC50 > 150 nM T54156 CO9QA4 44445209 IC50 = 88000 nM T54156 CH3UQ5 44445210 IC50 = 100000 nM T54156 C6B4LG 44445211 IC50 = 127000 nM T54156 C1WA5N 44445212 IC50 = 94000 nM T54156 CM2CD0 44445213 IC50 = 76000 nM T54156 C6ZX2P 44445214 IC50 = 50000 nM T54156 C9KE8P 44445215 IC50 = 3000 nM T54156 C68QEF 44445216 IC50 = 60000 nM T54156 CCK7W2 44445217 IC50 = 85000 nM T54156 C58BQA 44445218 IC50 = 71000 nM T54156 C4CGN2 44445219 IC50 = 33000 nM T54156 C1IVR6 44445220 IC50 = 67000 nM T54156 CG2U7H 44445221 IC50 = 69000 nM T54156 CVW48J 44445222 IC50 = 81000 nM T54156 CL3HZ8 44445223 IC50 = 68000 nM T54156 CPY73U 44445224 IC50 = 59000 nM T54156 C9MA2F 44445225 IC50 = 67000 nM T54156 C9SJM3 44445226 IC50 = 114000 nM T54156 CH91WG 44445228 IC50 = 73000 nM T54156 CO59HI 44445229 IC50 = 109000 nM T54156 C62WPE 44445230 IC50 = 103000 nM T54156 COIR35 44445231 IC50 = 114000 nM T54156 CBH0M7 44445233 IC50 > 150 nM T54156 CIS7M5 44445234 IC50 > 150 nM T54156 CKN60A 44445235 IC50 = 70000 nM T54156 CP4XL8 44445237 IC50 = 67000 nM T54156 CJA79R 44445239 IC50 = 90000 nM T54156 CA72BI 44445240 IC50 = 66000 nM T54156 CZJB48 44445241 IC50 = 132000 nM T54156 C85EVH 44445242 IC50 = 137000 nM T54156 C9DI7F 44445243 IC50 = 91000 nM T54156 CVLH67 44445244 IC50 = 88000 nM T54156 CIP3X8 44445245 IC50 = 107000 nM T54156 CL1MK6 44445246 IC50 = 112000 nM T54156 C0CX7T 44445247 IC50 = 7000 nM T54156 CEZ2P7 44445248 IC50 = 119000 nM T54156 CL0K9Q 44445249 IC50 = 126000 nM T54156 C9T2SH 44445250 IC50 = 141000 nM T54156 C5EFP9 44445251 IC50 = 93000 nM T54156 CLJ71G 44445252 IC50 = 95000 nM T54156 C8TF3E 44445253 IC50 = 83000 nM T54156 C4CAY7 44445254 IC50 = 107000 nM T54156 CH1LE5 44445255 IC50 = 120000 nM T54156 CLP96W 44445256 IC50 = 101000 nM T54156 CK8S4Z 44445257 IC50 = 140000 nM T54156 C03EJW 44445258 IC50 = 105000 nM T54156 CO9SM5 44445261 IC50 = 112000 nM T54156 C3FX8B 44445262 IC50 > 150000 nM T54156 CZS8N5 44445263 IC50 > 150000 nM T54156 CMW2U6 44445264 IC50 = 119000 nM T54156 CB47AH 44445265 IC50 = 150000 nM T54156 CA43LS 44445266 IC50 = 50000 nM T54156 C23MDF 44445267 IC50 = 75000 nM T54156 C9K3DI 44445268 IC50 = 110000 nM T54156 C2ZAK4 44445269 IC50 = 90000 nM T54156 CIVC64 44445270 IC50 = 109000 nM T54156 C8W1HX 44445271 IC50 > 150000 nM T54156 CTFR27 44445272 IC50 > 150000 nM T54156 C20DNO 44445273 IC50 > 150000 nM T54156 CWLC15 44445274 IC50 > 150000 nM T54156 CZD5M3 44445275 IC50 > 150000 nM T54156 CJET46 44445276 IC50 > 150000 nM T54156 CI58AM 44445277 IC50 > 150000 nM T54156 CDN37V 44445278 IC50 > 150000 nM T54156 CE36AB 44445279 IC50 > 150000 nM T54156 CV9KX5 44445280 IC50 > 150000 nM T54156 C4S2WX 44445281 IC50 > 150000 nM T54156 CP5H1Q 44446267 IC50 = 23 nM T54156 C30TQK 44446273 IC50 = 16400 nM T54156 CB76CO 44446275 IC50 = 24500 nM T54156 C20HIJ 44446753 IC50 = 111 nM T54156 C9CS8E 44446754 IC50 = 190 nM T54156 C4Z7IQ 44446755 IC50 = 110 nM T54156 C4K5QT 44446756 IC50 = 2500 nM T54156 C47SRV 44446758 IC50 > 5000 nM T54156 C8HM5N 44446763 IC50 > 5000 nM T54156 CU5Z4V 44446765 IC50 = 916 nM T54156 CYO65B 44446797 IC50 = 1268 nM T54156 CTKX08 44446807 IC50 = 604 nM T54156 CJN1L7 44446821 IC50 = 428 nM T54156 C4LF6Y 44446822 Ki = 934 nM T54156 C9FG5A 44446823 IC50 = 451 nM T54156 C1P0BV 44446824 IC50 = 309 nM T54156 C5AW3N 44446825 IC50 = 160 nM T54156 C17YSI 44446827 IC50 = 677 nM T54156 CE2OM1 44446839 IC50 = 2623 nM T54156 C49VJF 44446842 IC50 = 1499 nM T54156 CF4DL2 44446843 IC50 > 3000 nM T54156 CIP23G 44447330 IC50 = 1.7 nM T54156 CPS5M4 44447343 IC50 = 1.3 nM T54156 CB3F0E 44447344 IC50 = 0.89 nM T54156 CM7JV0 44447353 IC50 = 78 nM T54156 CY2XR5 44447363 IC50 = 86 nM T54156 CU2BC6 44447364 IC50 > 10000 nM T54156 CXS34M 44447371 IC50 = 29 nM T54156 CA5J9Q 44454525 IC50 > 10000 nM T54156 C6L1OH 44454554 IC50 = 104 nM T54156 CHTY64 44454555 IC50 = 54 nM T54156 CLNM62 44454612 IC50 = 39 nM T54156 CZ2QY4 44454641 IC50 = 54 nM T54156 C7DIB0 44454661 IC50 = 69 nM T54156 CTR91D 44454664 IC50 = 93 nM T54156 CR3PO9 44454741 IC50 = 933 nM T54156 C1ZSK0 44454742 IC50 = 242 nM T54156 CM8AG1 44454790 IC50 = 1489 nM T54156 CCH42M 44454856 IC50 = 984 nM T54156 CQG09B 44454861 IC50 = 6.6 nM T54156 CQ5YK3 44454864 IC50 = 31 nM T54156 CLG57Z 44454888 IC50 = 4819 nM T54156 CMEJ96 44454891 IC50 = 383 nM T54156 CV07DO 44455123 IC50 = 693 nM T54156 C9MHD2 44455124 IC50 = 57.9 nM T54156 C2L1VK 44455161 IC50 = 1.8 nM T54156 C4CZ7N 44455196 IC50 = 4.8 nM T54156 CZ15QG 44455197 IC50 = 32.6 nM T54156 CJ6L1K 44455200 IC50 = 1.3 nM T54156 CLK5O7 44455240 IC50 = 4.9 nM T54156 CSKN69 44455242 IC50 = 4.2 nM T54156 C3U9VM 44455265 IC50 = 33.4 nM T54156 CG65TZ 44455266 IC50 = 3.6 nM T54156 C14QTI 44455267 IC50 = 57.5 nM T54156 CSX4F2 44455294 IC50 = 4.4 nM T54156 CJ29BT 44455298 IC50 = 34.9 nM T54156 CCK15P 44455331 IC50 = 158.5 nM T54156 CW8IB7 44455332 IC50 = 1387 nM T54156 C9ZXF4 44455360 IC50 = 315 nM T54156 CFB78A 44455363 IC50 > 1000 nM T54156 CW46RV 44455498 Ki = 1851 nM T54156 CXNP45 44455499 Ki > 2128 nM T54156 C6CED5 44455528 Ki > 2128 nM T54156 CUQH30 44455553 Ki > 2128 nM T54156 C83KYJ 44455582 Ki > 2128 nM T54156 CK5N1S 44455612 Ki > 2128 nM T54156 CU2E7V 44455613 Ki > 2128 nM T54156 CH1DI4 44455614 Ki > 2128 nM T54156 CFQ79A 44455647 Ki > 2128 nM T54156 C3J1SV 44455676 IC50 = 21.1 nM T54156 CS6HL1 44455704 IC50 > 1000 nM T54156 CR4EX3 44455706 IC50 > 1000 nM T54156 CC01WS 44455737 IC50 = 846 nM T54156 C0R9SH 44455760 IC50 = 87.9 nM T54156 C6FV2Z 44455783 Ki > 2128 nM T54156 C7W6XV 44455786 IC50 = 13.9 nM T54156 CO58GJ 44455787 IC50 = 522 nM T54156 CPYV60 44455807 Ki > 2128 nM T54156 CLAT19 44455811 IC50 > 1000 nM T54156 C3TS1X 44455813 IC50 = 16.4 nM T54156 C92AFN 44455816 IC50 = 56.1 nM T54156 CGA0T4 44455829 Ki > 2128 nM T54156 CIR06N 44455835 IC50 = 45.8 nM T54156 C38VBL 44455836 IC50 = 7.3 nM T54156 CKB6E7 44455837 IC50 = 809 nM T54156 CV2B4N 44455858 Ki > 2128 nM T54156 CL6UY9 44455865 IC50 > 1000 nM T54156 CVR58Q 44455879 Ki > 2128 nM T54156 CWZ8K6 44455880 Ki > 2128 nM T54156 CD9N5I 44459425 Ki < 1 nM T54156 CP98IX 44459426 Ki < 1 nM T54156 CAM2Q6 44459443 Ki = 1.6 nM T54156 CM4T7A 44459538 Ki > 2128 nM T54156 CBNW98 44459546 Ki > 2128 nM T54156 CZ7LN0 44459591 Ki > 2128 nM T54156 C7YDK2 44459757 Ki > 2128 nM T54156 C1YQ7R 44459758 Ki = 2099 nM T54156 CI63AQ 44459833 Ki = 1490 nM T54156 CWEY79 44459834 Ki = 832 nM T54156 CA9DZ6 44459883 Ki = 1741 nM T54156 C09MZY 44459910 Ki = 1302 nM T54156 CEV0M3 44459911 Ki > 2128 nM T54156 CG0Z7I 44478924 IC50 = 410 nM T54156 CFO27Y 44478926 IC50 = 98 nM T54156 CBZJ29 44478927 IC50 = 94 nM T54156 CRJ24K 44479197 IC50 = 69 nM T54156 CGOH82 44479198 IC50 = 420 nM T54156 CLV56M 44479199 IC50 = 730 nM T54156 CY92OQ 44479458 IC50 = 51000 nM T54156 CH1QG9 44479459 IC50 = 930 nM T54156 CB1NT7 44479460 IC50 = 310 nM T54156 C0JQ9L 44479699 IC50 = 340 nM T54156 C0DN1Q 44479700 IC50 > 100000 nM T54156 CTG24W 44479702 IC50 = 20000 nM T54156 CGZ49M 44479703 IC50 = 3000 nM T54156 CAK94X 44563337 IC50 = 322 nM T54156 CJ2BU5 44563487 IC50 = 11 nM T54156 CP54WT 44563489 IC50 = 2563 nM T54156 C1UXP6 44563490 IC50 = 1246 nM T54156 CZ0W1A 44563491 IC50 = 732 nM T54156 C37UAM 44563492 IC50 = 827 nM T54156 C4BD0N 44563493 IC50 = 18 nM T54156 CR6NO2 44564180 IC50 = 23 nM T54156 CHQG04 44576676 Ki = 7900 nM T54156 CR65DO 44576708 Ki = 2.6 nM T54156 C2QFY7 44576710 Ki = 2750 nM T54156 C0BQV5 44576711 Ki = 150 nM T54156 CU2IP7 44576753 Ki = 1700 nM T54156 C8QHV1 44576806 Ki = 212000 nM T54156 C93LDF 44576807 Ki = 124000 nM T54156 C9T2KO 44576808 Ki = 150000 nM T54156 C7F3SX 44576850 Ki = 4200 nM T54156 CJ41MB 44576851 Ki = 329000 nM T54156 C9PUW2 44576877 Ki = 221000 nM T54156 CPT42K 44580109 IC50 > 5000 nM T54156 CQ7W5I 44580110 Ki < 1 nM T54156 CWD32S 44580184 IC50 = 5500 nM T54156 CQ4ZR1 44580422 IC50 = 560 nM T54156 C0XJ5C 44580496 Ki > 2128 nM T54156 CK68GT 44580539 Ki = 10.4 nM T54156 C2Z4HB 44583600 IC50 = 1788 nM T54156 C7PR8I 44583623 IC50 = 577 nM T54156 CDRC42 44583654 IC50 = 683 nM T54156 CM79HD 44583656 IC50 > 5000 nM T54156 CZNQ90 44593458 IC50 = 360 nM T54156 CTW7F2 44601281 IC50 = 8.7 nM T54156 C19LWR 44634267 IC50 = 2 nM T54156 CM0I4J 45101511 IC50 = 5000 nM T54156 CACH13 45269631 IC50 = 34 nM T54156 CH4NL1 45376336 IC50 = 1948.29 nM T54156 C3SQL2 45378250 IC50 = 190 nM T54156 CQE49A 45378251 IC50 = 1.1 nM T54156 CO4AC6 45378252 IC50 = 46 nM T54156 C42FPG 45378253 IC50 = 3.5 nM T54156 CI82BN 45378254 IC50 = 13 nM T54156 C6MY2W 45380188 IC50 = 170 nM T54156 C9P0DG 45380189 IC50 = 7.2 nM T54156 CRY0E8 45380190 IC50 = 8.6 nM T54156 C0MPH3 45380191 IC50 = 430 nM T54156 CMPE63 45482676 IC50 = 24000 nM T54156 C4ZWY7 45487310 IC50 = 5000 nM T54156 C9SV0H 45487311 IC50 = 5000 nM T54156 CCF05Q 45487333 IC50 = 498 nM T54156 CY09ZU 45487335 IC50 = 5000 nM T54156 COX40Y 45487358 IC50 > 5000 nM T54156 CF1T7M 45487359 IC50 = 5000 nM T54156 CRXI29 45487373 IC50 > 5000 nM T54156 CYL32E 45487376 IC50 > 5000 nM T54156 CO5P9I 45487386 IC50 > 5000 nM T54156 CS9Y8G 45487387 IC50 > 5000 nM T54156 CWLC18 45487393 IC50 > 5000 nM T54156 CI4KJ5 45487400 IC50 > 5000 nM T54156 C49HOI 45487401 IC50 = 5000 nM T54156 CSX5I9 46175170 IC50 = 58 nM T54156 C0S8FV 46231953 IC50 = 2300 nM T54156 CZ6C8P 46703060 IC50 = 5.91 nM T54156 C0DHL4 46703061 IC50 = 1753.85 nM T54156 CYA45K 46703062 IC50 = 3.64 nM T54156 CY72WL 46703063 IC50 = 5.67 nM T54156 C1YHS2 46703064 IC50 = 1632.42 nM T54156 C8HX7K 46840956 IC50 = 29270 nM T54156 CH0Z1E 46844314 Ki > 40000 nM T54156 C20BTY 46856241 Ki = 88400 nM T54156 C0ECU2 46861775 IC50 = 7.89 nM T54156 C0Y9NZ 46861793 IC50 = 7.29 nM T54156 C5L8GF 46871738 IC50 = 5000 nM T54156 CR1KF7 46871739 IC50 = 270 nM T54156 C8Q6YR 46871740 IC50 = 729 nM T54156 C58YSM 46871741 IC50 > 10000 nM T54156 C3X5EN 46873064 IC50 = 18320 nM T54156 CR3QW7 46891107 IC50 = 356 nM T54156 C5MK3A 46891108 IC50 = 2860 nM T54156 CQ5E1H 46891109 IC50 = 2090 nM T54156 C91LGI 46891170 IC50 = 163 nM T54156 CZPM12 46891172 IC50 = 722 nM T54156 C2V6MW 46891173 IC50 = 682 nM T54156 C8S7QX 46891209 IC50 > 10000 nM T54156 C5Y0MN 46891255 IC50 = 6700 nM T54156 CJ16SE 46891256 IC50 = 350 nM T54156 CNXU57 46891313 IC50 > 10000 nM T54156 CVK0E5 46891356 IC50 = 2501 nM T54156 C89RPO 46891357 IC50 > 10000 nM T54156 CVB6K4 46891358 IC50 > 10000 nM T54156 C0F7SU 46905989 IC50 = 101000 nM T54156 C49PYF 46907509 IC50 = 7.81 nM T54156 C2U1GW 46907510 IC50 = 8.19 nM T54156 C7MUS8 46907512 IC50 = 1869.59 nM T54156 C71YRF 46907513 IC50 = 1921.13 nM T54156 CVH58U 46907580 IC50 = 7.8 nM T54156 C0S9WB 46919610 Ki = 11000 nM T54156 CE3H7I 46938726 IC50 < 0.1 nM T54156 C9T0HR 46938727 IC50 = 0.18 nM T54156 C0YR7M 46938728 IC50 < 0.1 nM T54156 CUD7O0 50941549 IC50 > 10000 nM T54156 C5B6SP 50941565 IC50 = 11000 nM T54156 C7AU4S 50943150 IC50 > 100000 nM T54156 CAS94N 51346773 Ki = 3900 nM T54156 CP65WT 51346774 Ki = 12000 nM T54156 C5OIA2 51346775 Ki = 6200 nM T54156 CU2SX3 51355576 Ki > 10000 nM T54156 CLA96C 53232689 Ki = 430 nM T54156 C3BGW0 53233015 Ki > 40000 nM T54156 CZ06OY 53233469 IC50 = 2200 nM T54156 CMQZ70 53242178 IC50 > 25000 nM T54156 CRI92N 53311230 IC50 > 10000 nM T54156 C74CKF 53318123 Ki = 380 nM T54156 CTQ02K 53320639 IC50 = 460000 nM T54156 C4UE6R 53322469 IC50 > 100000 nM T54156 CI3WL5 53323418 Ki = 3500 nM T54156 CPY02U 53327890 IC50 = 63 nM T54156 CPGE80 53327891 IC50 = 77 nM T54156 CLJ4G2 53328858 IC50 = 79 nM T54156 C4G3QL 53328859 IC50 = 21 nM T54156 CX1TW0 53328860 IC50 = 4.3 nM T54156 C0ZX5G 53329215 IC50 = 50 nM T54156 CSU52A 53329216 IC50 = 650 nM T54156 CNB63X 53361475 IC50 = 22900 nM T54156 C6Y2EV 53374826 IC50 > 100000 nM T54156 CNY03Z 53378637 Ki = 3100 nM T54156 CX3DU4 53378973 Ki = 10000 nM T54156 CTD1H9 53378974 Ki = 9900 nM T54156 CBL30Y 54181369 IC50 > 10000 nM T54156 C3M8GZ 54580051 IC50 > 100000 nM T54156 CL0WM9 54580052 IC50 > 10000 nM T54156 CK26XF 54580053 IC50 > 10000 nM T54156 C3LF0P 54580544 Ki > 10000 nM T54156 CA8U9V 54580837 IC50 > 10000 nM T54156 C6R3MZ 54580973 Ki > 50000 nM T54156 CVO09J 54581546 Ki = 2400 nM T54156 CWB2Q6 54581896 IC50 = 670 nM T54156 CWKA42 54582019 Ki = 21000 nM T54156 CVK72M 54582073 IC50 = 3100 nM T54156 CBK18O 54582074 IC50 > 10000 nM T54156 CP2F1B 54582075 IC50 > 10000 nM T54156 CZNU23 54582076 IC50 > 10000 nM T54156 C0U5HZ 54582077 IC50 > 10000 nM T54156 C8SG9Y 54582079 IC50 > 10000 nM T54156 CZI6S3 54582080 IC50 > 10000 nM T54156 CD09BZ 54582543 IC50 = 1200 nM T54156 CH6Q2Z 54583016 IC50 > 10000 nM T54156 C3V9LQ 54583017 IC50 = 670 nM T54156 CT80KQ 54583018 IC50 > 1800 nM T54156 CPT4L5 54583019 IC50 > 10000 nM T54156 CK52YD 54583511 Ki = 1800 nM T54156 CF0SK8 54583712 IC50 = 23 nM T54156 CBEV27 54584024 IC50 > 10000 nM T54156 CM87DP 54584025 IC50 = 8500 nM T54156 C28GKQ 54585927 IC50 > 10000 nM T54156 CAZ76E 54586892 IC50 > 10000 nM T54156 CM0OQ3 54586893 IC50 > 10000 nM T54156 CK1NS7 54586894 IC50 > 10000 nM T54156 CMC4Y1 54586895 IC50 > 10000 nM T54156 C2MKX5 54586896 IC50 > 10000 nM T54156 CU91QP 54586897 IC50 > 10000 nM T54156 CI08RQ 54586898 IC50 = 1200 nM T54156 C6PRI4 54586899 IC50 = 8900 nM T54156 CG37UX 54587429 Ki = 1700 nM T54156 CL9SC3 54587769 Ki = 10100 nM T54156 C13FSJ 54669762 Ki = 870 nM T54156 CHS01Z 54669766 Ki = 19600 nM T54156 C8YLA4 54669829 IC50 = 1.9 nM T54156 C1KA8X 54669830 IC50 = 2.88 nM T54156 CZA6Q9 54669831 IC50 = 214 nM T54156 CF23NJ 54669841 IC50 = 87 nM T54156 C71KLJ 54679182 IC50 = 2520 nM T54156 C9P5ES 54752445 IC50 = 0.22 nM T54156 C0HKC9 54752446 IC50 = 0.58 nM T54156 C6D9IE 54753443 IC50 = 1819.27 nM T54156 CQD2Z6 54757100 IC50 = 611 nM T54156 C7E9SG 54757202 Ki = 490000 nM T54156 CMJ90D 54757404 Ki = 1600 nM T54156 CD1A3F 54757406 Ki = 4300 nM T54156 C4EFI5 54757409 Ki = 18700 nM T54156 C35BOE 56589587 IC50 = 25000 nM T54156 C5D1TI 56649332 IC50 = 7 nM T54156 CLKA98 56659256 IC50 = 43 nM T54156 CAFN81 56659257 IC50 = 1190 nM T54156 C5ATG7 56659258 IC50 = 173 nM T54156 CR0HX7 56659259 IC50 = 81 nM T54156 CG7E1O 56662736 IC50 = 13 nM T54156 CZF86Q 56662737 IC50 = 191 nM T54156 CT2G8L 56662738 IC50 = 25 nM T54156 C3LQY5 56662739 IC50 = 62 nM T54156 C8ZD7Q 56666204 IC50 = 43 nM T54156 CKB12J 56666205 IC50 = 45 nM T54156 CR21IL 56666206 IC50 = 77 nM T54156 CT65HD 56666207 IC50 = 74 nM T54156 C2IVE9 56666208 IC50 = 698 nM T54156 CC8HS0 56669604 IC50 = 28 nM T54156 CLO80F 56669605 IC50 = 70 nM T54156 CPS48C 56669606 IC50 = 376 nM T54156 CGMF96 56669607 IC50 = 51 nM T54156 CBX8M4 56673120 IC50 = 27 nM T54156 C6Z7VA 56673121 IC50 = 131 nM T54156 C2YJZ8 56673122 IC50 = 1.5 nM T54156 C3BD9S 56673123 IC50 = 198 nM T54156 CG10FP 56673124 IC50 = 978 nM T54156 CMNQ68 56673125 IC50 = 15 nM T54156 CWI28X 56676443 IC50 = 14 nM T54156 CSPX53 56676444 IC50 = 26 nM T54156 CJU1M7 56676445 IC50 = 19 nM T54156 CGD90C 56676446 IC50 = 282 nM T54156 CCA39I 56676447 IC50 = 57 nM T54156 C02GOU 56679764 IC50 = 16 nM T54156 CFDR70 56679765 IC50 = 14 nM T54156 CLPF34 56679766 IC50 = 36 nM T54156 C0XP1D 56679767 IC50 = 155 nM T54156 CTE68Z 56679768 IC50 = 34 nM T54156 CES0V3 56679769 IC50 = 93 nM T54156 CIB34L 56683087 IC50 = 5.2 nM T54156 CM79IH 56683088 IC50 = 1.1 nM T54156 CSL1X7 56683089 IC50 = 110 nM T54156 CSR32E 56683090 IC50 = 28 nM T54156 CWJ65H 56683091 IC50 = 215 nM T54156 CEO93F 56683092 IC50 = 120 nM T54156 CO8FP7 56683093 IC50 = 44 nM T54156 C6KT1Z 56683094 IC50 = 24 nM T54156 CJCI10 56683095 IC50 = 28 nM T54156 C5F7WT 56683096 IC50 = 80 nM T54156 C62FZC 56835063 IC50 = 1970 nM T54156 CKJ9S1 56835167 IC50 = 30 nM T54156 C21CLZ 56835168 IC50 = 660 nM T54156 C0L2TS 56835169 IC50 = 690 nM T54156 C8TH2F 56945850 IC50 = 9 nM T54156 CD72TG 56945851 IC50 = 4 nM T54156 C8J4SC 56945854 IC50 = 41 nM T54156 C1AIZ6 56945963 IC50 = 10 nM T54156 CXQC91 56945964 IC50 = 27 nM T54156 CM4H9D 56945965 IC50 = 74 nM T54156 CUT4S2 56946063 IC50 = 56 nM T54156 C2CQR8 56946064 IC50 = 23 nM T54156 C2H8PG 56946065 IC50 = 20 nM T54156 CW2P6A 56946167 IC50 = 7 nM T54156 CT8S3G 56946168 IC50 = 60 nM T54156 C6LR7O 56964014 IC50 = 91 nM T54156 CE12KU 56964015 IC50 = 152 nM T54156 CL42CX 56964110 IC50 = 212 nM T54156 C10BMZ 57127110 IC50 > 10000 nM T54156 CHE2I1 57345500 Ki > 50000 nM T54156 C63TFM 57345501 Ki > 50000 nM T54156 C8KT2F 57345502 Ki = 11000 nM T54156 C0KPD8 57384084 IC50 = 600 nM T54156 CV67JB 57384091 IC50 = 480 nM T54156 C5WFN6 57391082 IC50 = 2 nM T54156 C9BN4F 57391101 IC50 = 11 nM T54156 CN2H9K 57391204 IC50 > 10000 nM T54156 CR8MW2 57391205 IC50 > 10000 nM T54156 CAQB32 57391413 IC50 = 76000 nM T54156 CCB9H2 57391414 IC50 = 2 nM T54156 CC57MO 57392866 IC50 = 5.9 nM T54156 C4IWN7 57392867 IC50 = 1506 nM T54156 C1ZG3T 57392880 IC50 = 1 nM T54156 CNQ9B2 57392969 IC50 > 100000 nM T54156 CTYP14 57392972 IC50 > 10000 nM T54156 C5VB0U 57392973 IC50 > 10000 nM T54156 CMQL31 57392974 IC50 > 10000 nM T54156 C39OHF 57392975 IC50 > 10000 nM T54156 C0F3ZD 57393177 IC50 > 500000 nM T54156 CUJD65 57393178 IC50 = 430000 nM T54156 CMB13S 57393179 IC50 = 144000 nM T54156 CT2E8Z 57393181 IC50 > 50000 nM T54156 C2O9QP 57394596 IC50 = 1.3 nM T54156 CN9X5F 57394606 IC50 = 2 nM T54156 CP5BX6 57394607 IC50 = 11 nM T54156 CNOH63 57394711 IC50 > 10000 nM T54156 CE5X3D 57394850 IC50 = 5 nM T54156 C82ATC 57394900 IC50 = 30000 nM T54156 CG43ME 57394903 IC50 = 16 nM T54156 C18PVK 57396348 IC50 > 1000 nM T54156 CM8K2T 57396360 IC50 > 1000 nM T54156 CN0LI1 57396668 IC50 = 560 nM T54156 C2MI0H 57398136 IC50 = 1117 nM T54156 C98EXD 57398159 IC50 = 12 nM T54156 C1BIM8 57398160 IC50 = 16 nM T54156 C0KPT7 57398161 IC50 = 0.8 nM T54156 CD50CO 57399918 IC50 > 10000 nM T54156 C1CN3U 57401566 IC50 = 5091 nM T54156 C3EKY4 57401585 IC50 = 9 nM T54156 C2IE0C 57401902 IC50 = 47000 nM T54156 C39ELP 57403329 IC50 = 23 nM T54156 CWP09F 57403330 IC50 > 1000 nM T54156 CIB91W 57403331 IC50 = 0.21 nM T54156 C63WPS 57403332 IC50 = 0.2 nM T54156 CXF62Z 57403333 IC50 = 17 nM T54156 CK68EY 57403424 IC50 > 10000 nM T54156 C0G2VY 57403564 IC50 = 0.5 nM T54156 CE9B2P 57403620 IC50 = 1900 nM T54156 C1DRY0 57403621 IC50 = 230 nM T54156 C2MH8O 57523473 IC50 = 0.37 nM T54156 C57CEM 57523505 IC50 = 3 nM T54156 CS8W4L 57523538 IC50 = 2 nM T54156 CIT7B9 57523539 IC50 = 0.6 nM T54156 C56QXU 57523540 IC50 = 5 nM T54156 CX8IU3 57523541 IC50 = 43 nM T54156 CE8CL9 57523575 IC50 = 7 nM T54156 CWUP89 57523576 IC50 = 0.03 nM T54156 CT2QS3 57523577 IC50 = 0.06 nM T54156 CK6M0Y 57523578 IC50 = 0.05 nM T54156 C0HVU7 57523611 IC50 = 4 nM T54156 C5Q0ND 57523641 IC50 = 0.9 nM T54156 CWH7V8 57561293 IC50 = 1760 nM T54156 CY1N3J 57792153 IC50 = 1156 nM T54156 C6BKQ0 57874709 IC50 = 50000 nM T54156 CCKD80 58307579 Ki = 1.1 nM T54156 CX73PT 59033102 IC50 > 25000 nM T54156 CAT67H 59910477 IC50 = 4282 nM T54156 CTZJ24 59910497 IC50 = 7432 nM T54156 CLOE02 70682288 Ki = 290 nM T54156 CH2Q3V 70682301 IC50 = 47.58 nM T54156 C4NG7I 70682302 IC50 = 145 nM T54156 C6YOW4 70682303 IC50 = 12 nM T54156 CNM64E 70684016 IC50 = 197 nM T54156 CH76IU 70684364 Ki = 3000 nM T54156 CZ63AG 70684365 Ki = 470 nM T54156 C6YH8C 70684382 IC50 = 26 nM T54156 CQ50YR 70684390 IC50 = 97 nM T54156 CTR64D 70686538 IC50 = 92 nM T54156 C0Q6JA 70686539 IC50 = 104 nM T54156 C8B6WD 70688393 IC50 = 990 nM T54156 CGR3J2 70688394 IC50 = 21240 nM T54156 CX4M8O 70688395 IC50 = 9910 nM T54156 CTUN76 70688632 Ki = 44 nM T54156 C3LCG0 70688633 Ki = 160 nM T54156 CV9Y7S 70688643 IC50 = 8.1 nM T54156 CV2ZR4 70689156 IC50 = 1710 nM T54156 CJY19I 70690714 IC50 = 6.2 nM T54156 CFM0Q5 70690777 IC50 = 0.6 nM T54156 CWVI71 70691250 IC50 = 100 nM T54156 C8VTO0 70692397 IC50 = 2 nM T54156 C5AK0Y 70692405 IC50 = 0.5 nM T54156 CQ0D3Z 70692468 IC50 = 1.1 nM T54156 C1A0VU 70692840 Ki = 930 nM T54156 CY4E9Z 70692916 IC50 > 100000 nM T54156 CJGT23 70693360 IC50 = 360 nM T54156 C6P3XM 70693710 Ki > 50000 nM T54156 C0HE2P 70694634 IC50 = 3460 nM T54156 C51LCP 70695462 IC50 = 900 nM T54156 CENQ98 70697478 IC50 = 560 nM T54156 C1XNI9 70941086 IC50 = 100000 nM T54156 C7BHO9 70941091 IC50 = 100000 nM T54156 C37VPQ 70941121 IC50 = 8800 nM T54156 CF7PC5 70941155 IC50 = 100000 nM T54156 CL7JF9 71304794 IC50 = 26 nM T54156 CSY30R 71304795 IC50 = 5.5 nM T54156 CNPG78 71304796 IC50 = 510 nM T54156 CI8X5B 71449151 IC50 = 112 nM T54156 COM1B0 71449369 IC50 = 21 nM T54156 CD4CP2 71451167 IC50 = 19800 nM T54156 C6M9VL 71451168 IC50 = 27500 nM T54156 C7HUF5 71451169 IC50 = 86 nM T54156 CMW3O0 71451330 Ki = 148000 nM T54156 CGO17T 71452184 IC50 = 22 nM T54156 CE98YL 71452999 IC50 = 517 nM T54156 C8VC6N 71453000 IC50 = 170 nM T54156 C4VKI1 71453001 IC50 = 1800 nM T54156 C3KGU0 71453990 IC50 = 10 nM T54156 C9QS6E 71456659 Ki = 10 nM T54156 C04MJU 71457521 IC50 = 27 nM T54156 C2OL0I 71457963 IC50 = 410 nM T54156 CYB60V 71458014 IC50 = 230 nM T54156 CXC1U7 71458350 IC50 = 141 nM T54156 C4IZ5V 71458351 IC50 = 159 nM T54156 CU0Z4Y 71459396 IC50 = 1 nM T54156 CW7T3Y 71459397 IC50 = 1800 nM T54156 CHLW85 71459398 IC50 = 87 nM T54156 CZO86D 71460193 IC50 = 66 nM T54156 CU94ON 71461155 IC50 = 4500 nM T54156 CWL97M 71461905 IC50 = 103 nM T54156 CUT3H5 71461906 IC50 = 561 nM T54156 C06AXC 71461907 IC50 = 650 nM T54156 CSW59Y 71461908 IC50 = 3010 nM T54156 C29RWP 71462894 IC50 = 2 nM T54156 CATP87 71465323 IC50 = 3 nM T54156 C0H3BX 71465324 IC50 = 12.3 nM T54156 CTM24Y 71465370 IC50 = 4.9 nM T54156 C6ZV0X 71465371 IC50 = 8.3 nM T54156 C7NYO8 71465420 IC50 = 6.4 nM T54156 C0E3FD 71465421 IC50 = 0.54 nM T54156 CW1K8M 71465466 IC50 = 100000 nM T54156 C28OYX 71465467 IC50 = 100000 nM T54156 C12BUO 71465468 IC50 = 100000 nM T54156 CP37ZB 71465510 IC50 = 1700 nM T54156 CR2T8F 71503450 IC50 = 1.6 nM T54156 C8X0ST 71505576 IC50 = 1200 nM T54156 C56YRV 71516803 IC50 < 1 nM T54156 C52QIK 71516804 IC50 = 4.1 nM T54156 C79ZRK 71516805 IC50 < 1 nM T54156 C3L7SD 71533484 IC50 = 81 nM T54156 CZH5S9 71533485 IC50 = 222 nM T54156 C4YRC7 71533486 IC50 = 13 nM T54156 CGM72Q 71540498 IC50 = 85 nM T54156 CXA1I5 71540599 IC50 = 188 nM T54156 C7CV9E 71540600 IC50 = 115 nM T54156 CA4BP6 71540601 IC50 = 121 nM T54156 CMZ3T2 71540715 IC50 = 80 nM T54156 CXY83G 71540716 IC50 = 71 nM T54156 C1ZH2G 71540717 IC50 = 131 nM T54156 CT4UD5 71540831 IC50 = 120 nM T54156 CP7SX8 71540832 IC50 = 144 nM T54156 C9IW7R 71540833 IC50 = 50 nM T54156 C6MA8T 71540949 IC50 = 608 nM T54156 C52FXB 71547352 IC50 = 43.9 nM T54156 C9RE0A 71559535 IC50 = 7.57 nM T54156 C47TMN 71559652 IC50 = 7.63 nM T54156 CN2XB4 71559653 IC50 = 5.71 nM T54156 CZHQ79 71559654 IC50 = 1561.56 nM T54156 CO59LK 71559762 IC50 = 3.37 nM T54156 CGL35Z 71559763 IC50 = 5.82 nM T54156 C7U5LE 71559764 IC50 = 1658.63 nM T54156 CD6L1J 71559765 IC50 = 3.42 nM T54156 CXKO04 71559766 IC50 = 5.91 nM T54156 CA14SK 71559767 IC50 = 1758.72 nM T54156 COZ56A 71559768 IC50 = 8.02 nM T54156 CZ9X1J 71559769 IC50 = 1859.82 nM T54156 C5NHI1 71559770 IC50 = 7.79 nM T54156 CF9JE8 71559897 IC50 = 8.22 nM T54156 CGT96R 71559898 IC50 = 5.82 nM T54156 C01PTX 71559899 IC50 = 1585.79 nM T54156 C96OCB 71559900 IC50 = 5.91 nM T54156 CJB0D9 71559901 IC50 = 1659.85 nM T54156 C6Y1IE 71559902 IC50 = 4.32 nM T54156 C24ZYC 71559903 IC50 = 5.97 nM T54156 CC3MY7 71559904 IC50 = 1685.93 nM T54156 C7WMU5 71560026 IC50 = 8.93 nM T54156 C60VEX 71560027 IC50 = 1628.58 nM T54156 CN1VF7 71560028 IC50 = 8.41 nM T54156 CSY3D5 71560029 IC50 = 9.19 nM T54156 CH5J4A 71602247 IC50 = 107 nM T54156 CH53IU 71602248 IC50 = 3600 nM T54156 C97EWQ 71602249 IC50 = 1500 nM T54156 C7RZN9 71652216 IC50 = 96 nM T54156 CYS46I 71652677 IC50 = 6700 nM T54156 CX67VE 71654516 IC50 = 6000 nM T54156 C6KEH0 71680708 Ki = 210 nM T54156 C7DMX5 71680709 Ki = 15 nM T54156 CFPM82 71680710 Ki = 2.4 nM T54156 C9ZOM7 71680866 Ki = 3.6 nM T54156 CQ68LT 71680868 Ki = 30000 nM T54156 CFH2V0 71681183 Ki = 230 nM T54156 CV3X1T 71682766 Ki = 970 nM T54156 C5EAO8 71682767 Ki = 280 nM T54156 C80EYX 71682913 Ki = 9600 nM T54156 CIBD03 71682914 Ki = 630 nM T54156 C41BYG 71682915 Ki = 25 nM T54156 C93XEI 71682916 Ki = 42 nM T54156 CQ29PJ 71682917 Ki = 200000 nM T54156 CFWN65 71683062 Ki = 4300 nM T54156 CM4E5A 71716445 IC50 = 4.41 nM T54156 C45PSZ 71717046 IC50 = 9.34 nM T54156 C9Z4PI 71718276 IC50 = 7.52 nM T54156 C2XW5I 71718291 IC50 = 8.32 nM T54156 C18RDB 71719502 IC50 = 3.51 nM T54156 C6FVE5 71734008 IC50 = 1.1 nM T54156 CN95PL 71734104 IC50 = 11 nM T54156 CV37BJ 71734105 IC50 = 21 nM T54156 C7H8VM 71734106 IC50 = 97 nM T54156 CHBV73 71734107 IC50 = 460 nM T54156 C6C1JF 71734108 IC50 = 78 nM T54156 CR28AW 71734195 IC50 = 17 nM T54156 C2YJR3 71734196 IC50 > 1000 nM T54156 CJC6N5 71734197 IC50 = 38 nM T54156 CEF50T 71734198 IC50 = 100 nM T54156 CLWC38 72193198 IC50 < 1 nM T54156 CX4G0R 72204928 IC50 > 100000 nM T54156 CG9C6U 72204929 IC50 = 30000 nM T54156 C5A6XZ 72204930 IC50 = 20000 nM T54156 C0XZK4 72204931 IC50 > 100000 nM T54156 CM8Y7X 72204932 IC50 > 100000 nM T54156 C6RY4X 72204933 IC50 > 100000 nM T54156 C4N5AB 72204934 IC50 > 100000 nM T54156 C3H2FZ 72205111 IC50 > 100000 nM T54156 CQ0VX7 72205112 IC50 > 100000 nM T54156 CQ7TI1 72205113 IC50 > 100000 nM T54156 CPAW52 72205114 IC50 = 55000 nM T54156 C2LD3J 72205115 IC50 = 87000 nM T54156 CE4J8F 72711063 Ki = 860 nM T54156 CW2RF1 72711064 Ki = 1100 nM T54156 CC5T1Q 72711065 Ki = 2700 nM T54156 CTM4P2 72713638 IC50 = 1.4 nM T54156 C0N2JX 72713639 IC50 = 42 nM T54156 CF4K8Y 72713862 IC50 = 37 nM T54156 C3R6JO 72713863 IC50 = 690 nM T54156 CW9D3V 72713864 IC50 = 60 nM T54156 CQ6FH3 72713865 IC50 = 110 nM T54156 C4FYB0 72713866 IC50 = 76 nM T54156 CH6SI1 72713867 IC50 = 920 nM T54156 CS21QM 72713868 IC50 = 29000 nM T54156 CB56AP 72714081 IC50 = 330 nM T54156 C1CK0E 72714082 IC50 = 51000 nM T54156 COQZ24 72714091 Ki = 230 nM T54156 CC0ZX4 72714092 Ki = 930 nM T54156 CW8I1S 72714093 Ki = 1000 nM T54156 C3Q9LV 72714094 Ki = 1300 nM T54156 CZFY06 72714322 IC50 = 11000 nM T54156 CDY70J 72714323 IC50 = 4400 nM T54156 CD56BA 72714324 IC50 = 1630 nM T54156 CE51LQ 72714333 Ki = 12000 nM T54156 CK6D5F 72714334 Ki = 52000 nM T54156 C9FL7V 72714339 Ki = 180 nM T54156 CDX2F9 72984326 IC50 = 8.85 nM T54156 CTOQ24 73054451 IC50 > 100000 nM T54156 C9V6GC 73054734 IC50 > 100000 nM T54156 C63OXM 73054735 IC50 > 100000 nM T54156 CI14XA 73054736 IC50 > 100000 nM T54156 CK9TU0 73055013 IC50 = 1700 nM T54156 CFPC79 73055014 IC50 > 100000 nM T54156 C7UQ1B 73055016 IC50 > 100000 nM T54156 CO5FN4 73055018 IC50 > 100000 nM T54156 C8H0UN 73055605 IC50 > 100000 nM T54156 C01SHT 73055902 IC50 = 11000 nM T54156 C2GE8Q 73055903 IC50 = 9400 nM T54156 CDA75O 73055905 IC50 = 17000 nM T54156 CK5FT8 73055906 IC50 > 100000 nM T54156 C9OX6Y 73055907 IC50 = 16000 nM T54156 CA93JD 73056179 IC50 = 48000 nM T54156 CEX86T 73056180 IC50 = 50000 nM T54156 C8QZG6 73056181 IC50 > 100000 nM T54156 C1KGT9 73056183 IC50 > 100000 nM T54156 CR75BY 73056185 IC50 > 100000 nM T54156 C7YT0C 73056773 IC50 > 100000 nM T54156 CUKG79 73292708 IC50 = 6 nM T54156 C5D3CJ 73292709 IC50 = 4 nM T54156 CL69NM 73292710 IC50 = 4 nM T54156 CQ4RO1 73292711 IC50 = 0.07 nM T54156 C7CT2E 73292869 IC50 = 2 nM T54156 CA0LS6 73292870 IC50 = 0.3 nM T54156 CJU3V6 73292871 IC50 = 0.6 nM T54156 C3PGF2 73292872 IC50 = 3 nM T54156 C0O8VM 73292873 IC50 = 3 nM T54156 CBR9I5 73293034 IC50 = 0.4 nM T54156 C9FD2C 73293035 IC50 = 6 nM T54156 C7LP5J 73293036 IC50 = 2 nM T54156 C9PQG1 73293037 IC50 = 10 nM T54156 C4PF1H 73293038 IC50 = 0.8 nM T54156 CE39WF 73293196 IC50 = 3 nM T54156 CU96XE 73293197 IC50 = 11 nM T54156 CGC51Z 73293198 IC50 = 7 nM T54156 CC83FW 73293199 IC50 = 0.2 nM T54156 CS6T8M 73293200 IC50 = 0.2 nM T54156 C38IDL 73345835 Ki = 0.98 nM T54156 C25SOB 73349251 IC50 = 0.07 nM T54156 CW01EA 73349535 IC50 > 10000 nM T54156 C8ROG3 73350414 Ki = 5.7 nM T54156 CF7AB2 73350415 Ki = 4.9 nM T54156 C2PFM4 73351930 Ki = 5.3 nM T54156 CI09CY 73354906 Ki = 3.9 nM T54156 C7M4FT 74430862 IC50 = 25430 nM T54156 CUB7V9 76329513 IC50 = 1.4 nM T54156 C21FEO 76331549 IC50 = 174 nM T54156 CX39OW 76331563 IC50 = 399 nM T54156 C5LB0U 78426619 IC50 > 100000 nM T54156 CET6N8 78426757 IC50 > 100000 nM T54156 CKD41G 81689861 IC50 = 9000 nM T54156 CGQ8F3 86287515 IC50 = 10000 nM T54156 CJ37XE 86287516 IC50 = 17000 nM T54156 COV8I9 86291010 IC50 = 1210 nM T54156 CY74HT 89136066 IC50 = 4.6 nM T54156 C1MDQ8 89136114 IC50 = 700 nM T54156 CVPH63 90663059 Ki = 15000 nM T54156 C6AK3O 90663060 Ki = 14000 nM T54156 CUZD67 90663061 Ki = 10000 nM T54156 CTQ17J 90663062 Ki = 53000 nM T54156 CQGJ90 90663063 Ki = 2000 nM T54156 C0ZH1K 90663064 Ki = 14000 nM T54156 CD53CF 90663065 Ki = 4000 nM T54156 C1A4QT 90663067 Ki = 7000 nM T54156 CLW7Q8 90663069 Ki = 29000 nM T54156 C6JY4Q 90663070 Ki = 44000 nM T54156 C7YU1I 90663071 Ki = 17000 nM T54156 C07RTW 90663072 Ki = 5000 nM T54156 CZ68QM 90663073 Ki = 21000 nM T54156 CVTJ63 90663074 Ki = 5000 nM T54156 C9J8HB 90663075 Ki = 400 nM T54156 C06GRV 90663076 Ki = 300 nM T54156 CF2L9A 90663077 Ki = 50000 nM T54156 CGL0N7 90663078 Ki = 18000 nM T54156 COP05M 90663079 Ki = 10000 nM T54156 C1E5CB 90663080 Ki = 40000 nM T54156 C6IXP4 90663081 Ki = 45000 nM T54156 C0S7NT 90663082 Ki = 18000 nM T54156 C8MOY6 90663083 Ki = 20000 nM T54156 C4NP9W 90663084 Ki = 16000 nM T54156 CD3C8E 90663085 Ki = 15000 nM T54156 C63NOF 90663086 Ki = 21000 nM T54156 CU3LC2 90663087 Ki = 18000 nM T54156 CQ9C5I 90667651 IC50 = 0.53 nM T54156 CGXO89 90667652 IC50 = 0.32 nM T54156 CRT54C 101910871 IC50 = 65000 nM T54156 C1J3CK 117094707 IC50 = 24000 nM T54156 C1W5NH 118718816 IC50 = 1000 nM T54156 CDO15M 118721026 IC50 = 31.5 nM T54156 CHO72Q 118721027 IC50 = 2420 nM T54156 C4V3FD 118723755 IC50 = 346.4 nM T54156 CQ6C8V 121232412 IC50 = 1200 nM T54156 CH6OW5 122179777 IC50 = 40960 nM T54156 CLCW15 122181996 IC50 > 100000 nM T54156 CZO32N 122181998 IC50 > 100000 nM T54156 C40DWG 122181999 IC50 > 100000 nM T54156 CJFS09 122190237 IC50 = 3900 nM T54156 CRN56G 122191012 IC50 = 709.7 nM T54156 CGC3E2 122191014 IC50 = 833 nM T54156 CS61WU 122191016 IC50 = 677.2 nM T54156 CV3SP6 122191017 IC50 = 428.6 nM T54156 C8ZOT4 122191645 IC50 = 10890 nM T54156 CU6LT0 122191646 IC50 = 5430 nM T54156 CER90U 122191647 IC50 = 11970 nM T54156 C8X2BN 122191648 IC50 = 4290 nM T54156 CQ3US9 122191649 IC50 = 6720 nM T54156 C86DWE 122191650 IC50 = 7970 nM T54156 CQ14HT 122191651 IC50 = 12870 nM T54156 C8B1HC 122191652 IC50 = 15960 nM T54156 CN6WP3 122191653 IC50 = 1870 nM T54156 CJ5R2S 122192039 IC50 = 8610 nM T54156 CK45AP 122192040 IC50 = 3190 nM T54156 C2W4VX 122192041 IC50 = 5470 nM T54156 C3R5YP 122192042 IC50 = 33750 nM T54156 C8EB9C 122192043 IC50 = 7910 nM T54156 CF2K9Z 122192044 IC50 = 8720 nM T54156 C68DRB 122192045 IC50 = 5920 nM T54156 C2L7ZO 122192046 IC50 = 4680 nM T54156 C1BH0V 122192047 IC50 = 5960 nM T54156 C9MX4H 122192048 IC50 = 13890 nM T54156 CE4MD1 122192049 IC50 = 6910 nM T54156 CU13GZ 122192050 IC50 = 4950 nM T54156 CN1OP2 122192051 IC50 = 18960 nM T54156 C2WV6G 122192052 IC50 = 18310 nM T54156 CD2I6H 122192053 IC50 = 19810 nM T54156 CQ7RZ6 122192054 IC50 = 5880 nM T54156 C9FWL4 122195563 IC50 = 590 nM T54156 COIP89 122195564 IC50 = 60 nM T54156 C8Z1BF 124196387 IC50 > 1000000 nM T54156 C9QKI3 127020966 IC50 > 100000 nM T54156 CF9C4N 127025165 IC50 = 19 nM T54156 CH59PY 127025166 IC50 > 100000 nM T54156 CT03QA 127026888 IC50 = 4500 nM T54156 CO1DJ9 127027301 IC50 = 18.5 nM T54156 CM7B5S 127029507 IC50 = 393 nM T54156 C6HA8I 127029508 IC50 > 100000 nM T54156 CPM3N2 127029509 IC50 = 96.4 nM T54156 C3B9EY 127029510 IC50 > 100000 nM T54156 CV1YR6 127036461 IC50 = 2000 nM T54156 CDIC57 127037442 IC50 = 5.3 nM T54156 CV3NQ6 127037443 IC50 = 26000 nM T54156 CWI7K3 127037444 IC50 > 10000 nM T54156 C9QLI2 127037445 IC50 = 8200 nM T54156 CCA0R8 127037446 IC50 = 6200 nM T54156 C89QOM 127043503 IC50 = 6740 nM T54156 CK3I0F 127043504 IC50 = 2093 nM T54156 C9E5YJ 127043505 IC50 = 880 nM T54156 CW1Q3D 127043506 IC50 = 1155 nM T54156 CFDC75 127043682 IC50 = 1824 nM T54156 C1C7WB 127044036 IC50 = 7001 nM T54156 C16UNQ 127044037 IC50 = 5494 nM T54156 C5DMP0 127044039 IC50 = 5991 nM T54156 CPF6U7 127044139 IC50 = 11280 nM T54156 CT9B0Q 127044462 IC50 = 714.9 nM T54156 CL3X1A 127044649 IC50 = 8170 nM T54156 C7X1YO 127044650 IC50 = 8500 nM T54156 C8RZ7T 127044651 IC50 = 5715 nM T54156 C3I4PT 127044652 IC50 = 5882 nM T54156 CDX86T 127044818 IC50 = 636 nM T54156 C56OJV 127044819 IC50 = 492 nM T54156 CF7A5N 127044986 IC50 = 38449 nM T54156 CGLJ92 127045131 IC50 = 8710 nM T54156 C4HY6K 127045132 IC50 = 7407 nM T54156 C21LIW 127053364 IC50 = 1579.01 nM T54156 CR5VQ8 127053365 IC50 = 7.75 nM T54156 C19QXS 127053368 IC50 > 10000 nM T54156 CJ0G9N 127053369 IC50 > 10000 nM T54156 C2Q6UH 127053370 IC50 = 7297.04 nM T54156 CWM7U2 127053371 IC50 = 27.32 nM T54156 C1VRM8 127053372 IC50 = 155.19 nM T54156 CT76DR 127053375 IC50 = 13.52 nM T54156 CYA92R 130282633 IC50 = 2100 nM T54156 CO3QE2 130282636 IC50 = 2200 nM T54156 C4MB7N 132285189 Ki = 150 nM T54156 CTN42D 132941363 IC50 = 41000 nM T54156 C83FAY 134130294 Ki = 18 nM T54156 C4A1SP 134130575 Ki = 289 nM T54156 CT3G2U 134133460 IC50 = 2.5 nM T54156 C8VLY0 134144890 IC50 = 34 nM T54156 C93ZLI 134145328 IC50 = 41 nM T54156 CU24IK 134694685 IC50 = 1500 nM T54156 C7K4PA 135412054 IC50 > 100000 nM T54156 CHV2U1 135438561 IC50 > 10000 nM T54156 CN30DX 135438809 IC50 > 100000 nM T54156 C4FVJ1 135487604 IC50 = 50000 nM T54156 CSB0M9 135494223 IC50 = 19400 nM T54156 CV6IW1 135532303 IC50 = 17600 nM T54156 C1MOD4 135567320 IC50 > 10000 nM T54156 CN8YJ2 135960845 IC50 = 8000 nM T54156 CA5JR6 136054481 IC50 > 10000 nM T54156 CV47JN 136054485 IC50 = 2900 nM T54156 CZ48WO 136054487 IC50 > 10000 nM T54156 C8FGT0 136054495 IC50 = 1600 nM T54156 CG70BZ 136054516 IC50 = 5.3 nM T54156 CSM57W 136054520 IC50 = 72 nM T54156 CTY79S 136118013 Ki > 2128 nM T54156 CTE87J 136118014 Ki > 2128 nM T54156 CIEW62 136380958 IC50 = 36 nM T54156 C9HS7J 137287436 IC50 = 4.7 nM T54156 C4UMY5 137636781 IC50 > 5000 nM T54156 CR8H9Z 137644167 IC50 > 5000 nM T54156 CB8M6U 137646865 IC50 > 5000 nM T54156 CK4LE6 137647628 IC50 > 10000 nM T54156 C9CIY6 137651719 IC50 = 50 nM T54156 CZB75K 137657128 IC50 > 10000 nM T54156 CC3I9B 137660260 IC50 > 10000 nM T54156 CAB7Q6 137660566 IC50 > 10000 nM T54156 C4H0EM 137661370 IC50 > 5000 nM T54156 CZ8H6N 137661550 IC50 = 19000 nM T54156 C37HMX 137701229 Ki = 190 nM T54156 C1Q2BP 145949247 IC50 > 5000 nM T54156 C6TD4M 145949288 IC50 > 5000 nM T54156 CN9RD6 145949408 IC50 > 5000 nM T54156 C5FWA2 145949488 IC50 > 5000 nM T54156 CZS1N7 145949693 IC50 > 5000 nM T54156 C6IPV3 145949783 IC50 = 6800 nM T54156 CYG32L 145950058 IC50 > 5000 nM T54156 C72LGN 145950074 IC50 = 7500 nM T54156 CU53BP 145950331 IC50 > 5000 nM T54156 CY8C4A 145950332 IC50 > 5000 nM T54156 CAJ25P 145951291 IC50 > 5000 nM T54156 C3EF7N 145952515 IC50 > 5000 nM T54156 CW1GS2 145952760 IC50 > 5000 nM T54156 CFN1R7 145952843 IC50 > 5000 nM T54156 CM6T2O 145953417 IC50 > 5000 nM T54156 C6FYK8 145953609 IC50 > 5000 nM T54156 CV80WQ 145954107 IC50 > 5000 nM T54156 C16VNH 145954604 IC50 > 5000 nM T54156 CQF50V 145954863 IC50 > 5000 nM T54156 C2HAG8 145955226 IC50 = 5140 nM T54156 C8QW9G 145955776 IC50 > 5000 nM T54156 CH0ZO5 145955778 IC50 > 5000 nM T54156 CFDZ62 145955866 IC50 > 5000 nM T54156 CVZ5U7 145955868 IC50 > 5000 nM T54156 C8TPR1 145956198 IC50 > 5000 nM T54156 COR96H 145956298 IC50 = 5970 nM T54156 CR8U7Y 145956318 IC50 > 5000 nM T54156 C7R3FE 145956426 IC50 = 7000 nM T54156 C4S8LU 145956764 IC50 > 5000 nM T54156 CUS0Y9 145957234 IC50 > 5000 nM T54156 CUO69Q 145957392 IC50 > 5000 nM T54156 CX94UK 145957493 IC50 > 5000 nM T54156 C6MHN7 145957508 IC50 > 5000 nM T54156 CQ15DP 145957734 IC50 = 6360 nM T54156 C5K7PV 145958060 IC50 > 5000 nM T54156 CBE02W 145958354 IC50 > 5000 nM T54156 CQL4O0 145959327 IC50 > 5000 nM T54156 CG03OE 145959777 IC50 = 6370 nM T54156 CIQ9J2 145960035 IC50 = 4800 nM T54156 CUAT97 145960347 IC50 > 5000 nM T54156 CZ76WA 145962290 IC50 > 5000 nM T54156 C27MTZ 145962695 IC50 > 5000 nM T54156 CRY63E 145963538 IC50 > 5000 nM T54156 CVCL61 145963739 IC50 > 5000 nM T54156 C8UC1T 145963891 IC50 > 100000 nM T54156 CWOF29 145964116 IC50 = 72600 nM T54156 CKD86B 145964366 IC50 = 56200 nM T54156 CI0T9C 145964617 IC50 = 66600 nM T54156 C3MDU9 145965508 IC50 = 36010 nM T54156 CA94UB 145966060 IC50 = 34800 nM T54156 CL7QD9 145966162 IC50 = 54600 nM T54156 C8M7FR 145966330 IC50 = 2960 nM T54156 CA80DF 145966420 IC50 = 83400 nM T54156 CNR98O 145966867 IC50 = 36300 nM T54156 C5ICD0 145967022 IC50 = 14300 nM T54156 CI9JB5 145967177 IC50 = 93100 nM T54156 CJ47BV 145969859 IC50 = 51900 nM T54156 C1R9ES 145971386 IC50 = 27400 nM T54156 CFE1A5 145971595 Ki = 19 nM T54156 CWY5X0 145971805 IC50 = 1430 nM T54156 CQ78MP 145971807 IC50 > 100000 nM T54156 CX0JY3 145972073 IC50 > 100000 nM T54156 C1FPG2 145972660 IC50 > 5000 nM T54156 CPB91X 145972781 IC50 = 8800 nM T54156 CQ4K0X 145972990 IC50 > 100000 nM T54156 CYFI60 145973042 IC50 = 24500 nM T54156 CG4E3F 145973485 IC50 = 51600 nM T54156 CJF73O 145973630 IC50 > 5000 nM T54156 CTA0S4 145974193 IC50 = 24300 nM T54156 C52HKA 145974836 IC50 = 43900 nM T54156 CKW8B6 145975533 IC50 = 48300 nM T54156 CV9D1F 145975682 IC50 = 24690 nM T54156 CTD40B 145975699 IC50 > 100000 nM T54156 CMNS71 145975707 IC50 = 20900 nM T54156 CI9VB4 145975902 IC50 > 10000 nM T54156 CM6QB0 145976230 IC50 > 100000 nM T54156 CU7HO6 145976282 IC50 = 57800 nM T54156 CW6F2Y 145976412 IC50 = 53600 nM T54156 CX7M9L 145976456 IC50 > 5000 nM T54156 C5C6VJ 145976464 IC50 > 100000 nM T54156 C1KPL5 145976497 IC50 = 5800 nM T54156 C18OCA 145976989 IC50 = 332000 nM T54156 CBD28P 145977013 IC50 > 100000 nM T54156 CPD1B0 145977213 IC50 > 5000 nM T54156 C8CV6O 145977231 IC50 > 100000 nM T54156 C3VOQ8 145978127 IC50 = 95900 nM T54156 C9Z5DX 145978402 IC50 > 5000 nM T54156 C2JQ6E 145978441 IC50 = 33600 nM T54156 C8ZVJ6 145978450 IC50 = 82600 nM T54156 C42JOA 145978615 IC50 > 100000 nM T54156 CFP7Q1 145979987 IC50 = 880 nM T54156 CB2J6O 145980521 IC50 > 50000 nM T54156 CLK6W4 145980984 IC50 = 520 nM T54156 C0OV4I 145982041 IC50 = 1120 nM T54156 C5Z7XW 145983264 IC50 = 242 nM T54156 C0EMZ9 145984335 IC50 = 388 nM T54156 CBNO84 145985441 IC50 = 524 nM T54156 CDW7K5 145986213 IC50 = 162 nM T54156 CX15IY 145986836 IC50 = 1235 nM T54156 C1TSJ5 145987118 IC50 = 2200 nM T54156 CC82EI 145987827 IC50 = 32 nM T54156 CNR3F4 145991781 IC50 = 890 nM T54156 C89PNI 145992859 IC50 = 5400 nM T54156 CT7BR3 145994093 IC50 = 2600 nM T54156 CM7YB8 145998092 IC50 > 100000 nM T54156 C2CZ9B 155511425 IC50 = 5100 nM T54156 CZ25LW 155512044 IC50 = 64000 nM T54156 CV10AF 155512426 IC50 = 845 nM T54156 C1V4CS 155512637 IC50 > 10000 nM T54156 CMQ8W6 155512861 IC50 > 10000 nM T54156 CFHU79 155514943 IC50 = 1000 nM T54156 C13OQY 155515143 IC50 = 5300 nM T54156 CC15YH 155515706 IC50 > 10000 nM T54156 C98HMU 155515777 IC50 = 1.25 nM T54156 C6N3DB 155517141 IC50 = 0.91 nM T54156 CF64GH 155518335 Ki = 2588 nM T54156 CS6ZT7 155519964 IC50 = 47 nM T54156 CG2RF3 155520398 IC50 > 100000 nM T54156 CL16UE 155520835 IC50 > 10000 nM T54156 C5C1SL 155521791 IC50 > 10000 nM T54156 C59YHT 155522902 IC50 = 731 nM T54156 C4AH9W 155525335 IC50 > 10000 nM T54156 CM9AP3 155526116 IC50 > 10000 nM T54156 C83IXL 155528558 IC50 = 0.76 nM T54156 CT4PA7 155528661 IC50 > 10000 nM T54156 CWB4X1 155529076 IC50 > 10000 nM T54156 CSG54J 155529234 IC50 > 10000 nM T54156 C2G0BE 155529579 IC50 > 10000 nM T54156 CC5FA9 155529859 IC50 > 10000 nM T54156 CQUA53 155531128 IC50 > 10000 nM T54156 C7TP3R 155531151 IC50 > 10000 nM T54156 CZSY48 155533962 IC50 = 1700 nM T54156 CG47PB 155534833 IC50 = 3600 nM T54156 C4DSL8 155536899 IC50 > 10000 nM T54156 CNH2K4 155540729 IC50 = 3500 nM T54156 CRY3D4 155541376 IC50 = 14 nM T54156 CJN8X5 155542058 Ki = 2.6 nM T54156 CO8ZY9 155542845 IC50 = 35 nM T54156 C1VL8X 155544079 IC50 > 10000 nM T54156 CYK18P 155544623 IC50 > 10000 nM T54156 CWEG57 155545190 IC50 = 120 nM T54156 CP6W3Q 155545205 IC50 > 10000 nM T54156 COH0W2 155546374 IC50 = 4370 nM T54156 CLT8Z2 155546617 IC50 = 520 nM T54156 C3FRY8 155547834 IC50 = 0.122 nM T54156 C1FP0M 155548067 IC50 = 1800 nM T54156 C9AOK6 155550135 IC50 > 10000 nM T54156 C9BW6U 155551066 IC50 = 1390 nM T54156 C9ZUH8 155553520 IC50 > 10000 nM T54156 CPQ84I 155553728 IC50 > 10000 nM T54156 C94NQE 155556307 IC50 > 10000 nM T54156 C9FC1W 155557598 IC50 = 2100 nM T54156 CG2DI6 155560100 IC50 > 10000 nM T54156 CQJ07L 155561559 IC50 = 6000 nM T54156 C3BA9L 155561798 IC50 = 108 nM T54156 CH40UO 155562232 IC50 = 2.1 nM T54156 C6SAE0 155562336 IC50 = 22 nM T54156 CD18KU 155563750 IC50 = 3100 nM T54156 CM0LN1 155563771 IC50 = 1300 nM T54156 C29SMF 155565303 IC50 > 10000 nM T54156 C51ZMC 155565586 IC50 = 660 nM T54156 CZ0WK1 155566979 IC50 = 3200 nM T54156 CU42CE 155567829 IC50 > 100000 nM T54156 C8D5VK 155567855 IC50 = 14000 nM T54156 CHL0F3 155567858 IC50 > 10000 nM T54156 C5U9LI 155569346 IC50 = 4000 nM T54156 CLT4Y6 10138589 Ki = 130 nM T54156 C5U3AO 57394286 IC50 = 7 nM T54156 D00RNA 44446270 IC50 = 1410 nM T54156 D00TRF 44423683 IC50 = 256000 nM T54156 D01UNE 44580457 Ki = 35.6 nM T54156 D02ADV 594397 IC50 > 10000 nM T54156 D02ECA 448942 IC50 = 980 nM T54156 D02EFQ 10549609 IC50 = 1500 nM T54156 D03AMR 9849669 Ki = 5 nM T54156 D03QAN 71166 IC50 = 100000 nM T54156 D03SNK 644601 IC50 = 14000 nM T54156 D03WJG 9910222 Ki = 0.06 nM T54156 D04GOO 10111838 IC50 > 100000 nM T54156 D04PAW 16216218 IC50 = 15000 nM T54156 D04VPH 45376872 IC50 = 8900 nM T54156 D04WWO 9889867 Ki > 2128 nM T54156 D05BMD 44423684 IC50 = 261000 nM T54156 D05THD 44478925 IC50 = 7700 nM T54156 D06EHW 11625778 IC50 = 304 nM T54156 D06HSC 136117931 IC50 = 22000 nM T54156 D06NDR 44423687 IC50 = 125000 nM T54156 D07DRT 46175162 Ki = 1.5 nM T54156 D07GEL 10344307 Ki = 0.9 nM T54156 D07MJD 44479701 IC50 = 7300 nM T54156 D07SPC 24857837 Ki = 227 nM T54156 D07VXX 16721024 IC50 = 352000 nM T54156 D08ICI 44446277 IC50 = 5660 nM T54156 D09GIL 66160 IC50 = 11000 nM T54156 D09GLA 4368 IC50 = 5 nM T54156 D09USO 5277466 IC50 > 100000 nM T54156 D09ZOA 25049753 IC50 = 34 nM T54156 D0A0FY 44479457 IC50 = 24000 nM T54156 D0A4TC 446504 IC50 = 4.3 nM T54156 D0A5MV 11581319 IC50 = 5410 nM T54156 D0B3UN 44580458 Ki = 1265 nM T54156 D0E5MB 44411812 IC50 = 10005 nM T54156 D0G0OP 44423685 IC50 = 141000 nM T54156 D0G3YZ 11391583 IC50 = 16500 nM T54156 D0H6CK 10160968 Ki > 2128 nM T54156 D0J5VK 67145 IC50 = 43400 nM T54156 D0K4TI 49292 IC50 = 330 nM T54156 D0L4EO 11609208 IC50 = 3600 nM T54156 D0L6ND 10089677 IC50 = 0.79 ug.mL-1 T54156 D0NP8A 10370504 IC50 = 840 nM T54156 D0NV9C 22004198 IC50 = 290 nM T54156 D0P2TS 9818682 IC50 > 10000 nM T54156 D0Q4TA 10044321 IC50 = 200 nM T54156 D0Q9LC 44385624 IC50 = 863 nM T54156 D0R2BO 194777 IC50 = 0.38 nM T54156 D0S9OL 10155934 IC50 = 690 nM T54156 D0T1FR 44457233 IC50 = 20000 nM T54156 D0V9EN 689043 IC50 = 21.22 nM T54156 D0V9GS 651854 IC50 = 160 nM T54156 D0W2UK 6914621 Ki = 10340 nM T54156 D0XK7G 10445302 IC50 = 130 nM T54156 D0XL8K 44313734 IC50 = 10.4 nM T54156 D0Y1XM 44423686 IC50 = 81000 nM T54156 D0Y5IQ 44255320 IC50 = 5000 nM T54156 D0Y7NV 2220392 IC50 = 696 nM T54156 D0Z4LO 9832179 IC50 = 7 nM T76937 D03FLC 3878 IC50 = 17000 nM T76937 D08HQK 5411 IC50 = 740 nM T76937 D0C7ET 11174599 IC50 = 5.3 nM T76937 D0X4RN 3676 IC50 = 10500 nM T76937 D00BUR 216327 IC50 > 1000 nM T76937 D04JZH 11659955 IC50 = 14000 nM T76937 D0K9IF 71666749 IC50 > 30000 nM T76937 D0O7QA 46840946 IC50 > 10000 nM T76937 D0OX9F 16046068 IC50 = 23000 nM T76937 CPN25U 998021 IC50 < 20 nM T76937 CXP8J4 1548400 IC50 = 3790 nM T76937 C2LSV1 15951112 IC50 = 2506 nM T76937 C8Q5MV 16039758 IC50 = 45 nM T76937 CK5GF0 25138300 IC50 = 155 nM T76937 CP72MB 25159060 IC50 = 10000 nM T76937 C01MRG 44603427 IC50 < 2000 nM T76937 CKW2T6 45102590 IC50 = 20 nM T76937 C40BIM 45139151 IC50 = 11 nM T76937 CS5EJ1 46841648 IC50 > 10000 nM T76937 CRE97F 46841787 IC50 > 10000 nM T76937 C06OXV 52920492 IC50 = 22000 nM T76937 CMS2F7 53239561 IC50 = 4760 nM T76937 C23WVS 53361524 IC50 = 300 nM T76937 CZO3W0 57732195 IC50 = 147 nM T76937 CCQ20P 59432866 IC50 = 1273 nM T76937 CYF3R7 60167367 IC50 = 12000 nM T76937 CT1YQ7 68680505 IC50 = 6900 nM T76937 C2MC6B 71522734 IC50 = 9330 nM T76937 CZ8KG6 71716851 IC50 = 30 nM T76937 C9MUK3 71716856 IC50 = 292 nM T76937 CUG2V3 71716866 IC50 > 3000 nM T76937 C7OE1X 76309796 IC50 = 24000 nM T76937 CBH4N7 76309797 IC50 = 28000 nM T76937 C10UTF 76310404 IC50 > 30000 nM T76937 C6T1NV 76310406 IC50 > 30000 nM T76937 CC4BK5 76310408 IC50 > 30000 nM T76937 C8M7RN 76310409 IC50 > 30000 nM T76937 CHFC49 76313502 IC50 > 30000 nM T76937 C1PM7H 76314065 IC50 > 30000 nM T76937 CBK0T8 76314067 IC50 > 30000 nM T76937 C20ILA 76314069 IC50 = 22000 nM T76937 C8OQT1 76314070 IC50 = 25000 nM T76937 CNM4K0 76317019 IC50 > 30000 nM T76937 C32OSF 76317020 IC50 = 27000 nM T76937 CKG5A9 76317629 IC50 > 30000 nM T76937 CQ7JK4 76317631 IC50 = 8000 nM T76937 CT2R5J 76320732 IC50 > 30000 nM T76937 CVP8U9 76320733 IC50 = 25000 nM T76937 C2RJW0 76320734 IC50 = 26000 nM T76937 CY8NT4 76321352 IC50 > 30000 nM T76937 CRU30A 76321353 IC50 = 13000 nM T76937 C46MFT 76324385 IC50 = 16000 nM T76937 C4W1NV 76324386 IC50 = 26000 nM T76937 CJF20G 76324950 IC50 = 27000 nM T76937 CP3UI7 76327945 IC50 > 30000 nM T76937 CNY5X1 76328517 IC50 = 23000 nM T76937 CX54MA 76328518 IC50 = 25000 nM T76937 CINA95 76331591 IC50 = 20000 nM T76937 CCXK29 76332197 IC50 > 30000 nM T76937 CH4K7Q 76332198 IC50 = 12000 nM T76937 C4WO6Y 76332199 IC50 = 27000 nM T76937 CK47NO 76332200 IC50 = 26000 nM T76937 CANB89 76332201 IC50 = 25000 nM T76937 CO2N7R 76335221 IC50 > 30000 nM T76937 C05RSQ 76335223 IC50 = 18000 nM T76937 C8ND6L 76335224 IC50 = 26000 nM T76937 CUO84S 76335833 IC50 > 30000 nM T76937 CTG76E 86687532 IC50 = 21000 nM T76937 CG2S4W 87487300 IC50 = 4450 nM T76937 CET9C7 87488556 IC50 = 197 nM T76937 CC5N9I 117737142 IC50 > 14000 nM T76937 C10BKY 117749324 IC50 > 42500 nM T76937 C9KV7L 117993993 IC50 = 12500 nM T76937 C7HJ6B 118126600 IC50 = 3500 nM T76937 C7AYV5 118540795 IC50 = 6400 nM T76937 CR8TX9 118708662 IC50 = 25 nM T76937 C9JL4Y 118937760 IC50 = 7100 nM T76937 C9Q2ND 121333973 IC50 = 6900 nM T76937 C9K5RV 122513516 IC50 > 20000 nM T76937 C09QIY 127047645 IC50 = 3400 nM T76937 CZ5H2B 132020452 IC50 > 30000 nM T76937 CFA52O 145979095 IC50 = 851 nM T76937 C30NUX 145979170 IC50 = 1640 nM T76937 C7O8DB 145979583 IC50 = 959 nM T76937 CJ2L1N 145982155 IC50 = 6675 nM T76937 CZN0U6 145982478 IC50 = 22 nM T76937 CQ9L7O 145987103 IC50 = 945 nM T76937 C8Q2EG 145988110 IC50 = 13 nM T76937 CT0Q9C 145989016 IC50 = 160 nM T76937 C7LGP9 145989565 IC50 = 296 nM T76937 C3YU9F 145990047 IC50 = 1830 nM T76937 CSPX23 145990181 IC50 = 993 nM T76937 C81UEC 145990738 IC50 > 3000 nM T76937 C9S1TW 145991701 IC50 = 374 nM T76937 C18AXJ 145992585 IC50 = 1955 nM T76937 C3N9FT 145992777 IC50 = 522 nM T76937 C4EFH0 145993219 IC50 = 124 nM T76937 CY7G9A 145993317 IC50 = 1793 nM T76937 CNF74P 145993643 IC50 > 3000 nM T76937 C2Z6DL 145994290 IC50 = 237 nM T76937 CG6OC3 155511866 IC50 = 110 nM T76937 CZ7X5M 155522127 IC50 = 15700 nM T76937 CCQ9Y1 155533815 IC50 = 260 nM T76937 C5ETZ0 155540932 IC50 = 200 nM T76937 CE3H4Z 155567528 IC50 = 210 nM T76937 D0FF6S 16038374 IC50 = 2450 nM T76937 D0P8TL 56947150 IC50 = 13 nM T11211 D06CNP 9821849 EC50 = 17050 nM T11211 D06XMU 6013 EC50 = 1.1 nM T11211 D07BSQ 5994 Ki = 8.5 nM T11211 D07MCK 5147 IC50 > 1000 nM T11211 D08QMX 5757 IC50 = 19.1 nM T11211 D0B2WJ 3371 IC50 > 50000 nM T11211 D0BC2E 91649 Ki = 2 nM T11211 D0D1SG 5755 IC50 > 2000 nM T11211 D0EP0C 5833 Ki = 39.4 nM T11211 D0G8BV 6450278 Ki = 315 nM T11211 D0IT2G 5743 IC50 > 1000 nM T11211 D0L2LS 6446 EC50 = 0.3 nM T11211 D0M1YR 15951529 Ki = 28.2 nM T11211 D0Q4SD 443872 IC50 > 10000 nM T11211 D0R1RS 3715 EC50 = 0.14 nM T11211 D0S6JG 5920 IC50 > 50000 nM T11211 D0S7LG 24872560 IC50 = 16 nM T11211 D0SN9T 4493 IC50 = 9 nM T11211 D0T2PL 5280453 IC50 > 10000 nM T11211 D0V9BD 2375 Ki = 19 nM T11211 D0Y0SW 3397 IC50 = 154 nM T11211 D0Z4EI 55245 Ki = 0.65 nM T11211 D00JFE 56941241 IC50 > 4000 nM T11211 D01SYU 10026128 IC50 = 10000 nM T11211 D03CVT 77461273 Ki = 18.4 nM T11211 D07MON 5311505 Ki > 100 nM T11211 D08AAV 46893585 IC50 = 1778.28 nM T11211 D08TEJ 11750009 Ki = 40 nM T11211 D09ZLZ 44200882 EC50 = 0.1 nM T11211 D0B4VE 10251 IC50 = 20000 nM T11211 D0HE7C 134415769 IC50 = 484 nM T11211 D0J6XC 5803 IC50 = 34800 nM T11211 D0L3HU 6918548 IC50 = 54 nM T11211 D0L4FS 5280961 IC50 = 1300000 nM T11211 D0LI1C 44469321 IC50 > 30000 nM T11211 D0NE3W 11326715 IC50 = 3.8 nM T11211 D0RV6F 11950726 EC50 = 144 nM T11211 D0SZ1G 121248172 IC50 > 100000 nM T11211 D0U0BU 11188409 EC50 = 405 nM T11211 D0X1OW 86287635 IC50 = 30000 nM T11211 D0DK4I 4534 IC50 = 38800 nM T11211 D0E2TY 71523527 EC50 = 0.14 nM T11211 D0M6LX 56851703 IC50 = 4700 nM T11211 D0O4QB 3314 IC50 = 19054.61 nM T11211 D0TH6M 25204767 EC50 > 10000 nM T11211 D02KAU 46871935 IC50 > 8910 nM T11211 D03KTE 16750192 Ki = 1.5 nM T11211 D08DZZ 10634 IC50 = 212 nM T11211 D0L5KF 132981 IC50 = 32 nM T11211 D0W5RL 9577221 IC50 = 9 nM T11211 C59UQE 6279 Ki = 2.9 nM T11211 C0XDJ1 9880 Ki = 14 nM T11211 C5NLY9 21648 IC50 = 251188.64 nM T11211 CTI9C4 31211 IC50 = 151356.12 nM T11211 C8ODZ3 56069 Ki = 10 nM T11211 C6I9HU 97860 IC50 = 39500 nM T11211 CB1A2Y 100790 IC50 = 1 nM T11211 CU0C6S 131698 EC50 = 9500 nM T11211 C1YH0B 161860 IC50 < 1000 nM T11211 CPW0V2 165521 IC50 = 851.14 nM T11211 CBR03V 173273 IC50 = 260 nM T11211 C0X8NW 176925 IC50 < 1000 nM T11211 C70YVR 179999 IC50 > 10000 nM T11211 C4DPB7 194069 IC50 = 28 nM T11211 C9NR7Q 242062 IC50 > 10000 nM T11211 CIG20C 243118 IC50 = 310 nM T11211 CDHI70 251929 IC50 = 40 nM T11211 CJMB61 256659 IC50 = 5900 nM T11211 CDP78A 261349 IC50 = 2250 nM T11211 CDM60I 261393 IC50 = 776.25 nM T11211 C0XDJ5 371219 IC50 > 10000 nM T11211 CNZ5P3 576549 IC50 > 200000 nM T11211 C8Y7MQ 610479 IC50 = 47000 nM T11211 CS1T2J 673702 IC50 = 9160 nM T11211 C2B0JA 674359 Ki = 7400 nM T11211 C2TX1C 676288 IC50 = 6190 nM T11211 C0JHO4 683402 IC50 = 650 nM T11211 C3GX7A 693178 IC50 = 510 nM T11211 C97LZN 693179 IC50 = 840 nM T11211 CF8YH9 727584 IC50 = 280 nM T11211 C2C4OW 737588 IC50 = 5050 nM T11211 CQ46YC 738483 IC50 = 630 nM T11211 C7U5YF 738487 IC50 = 1270 nM T11211 C69IAF 752037 IC50 = 7400 nM T11211 C7W1JQ 760603 IC50 = 4600 nM T11211 C1B3RI 760604 IC50 = 11100 nM T11211 CIJO46 761631 IC50 = 18640 nM T11211 CIGA96 794157 IC50 = 33400 nM T11211 CRT6Y4 802764 IC50 = 1660 nM T11211 C5MS0Y 843205 IC50 = 3760 nM T11211 C61ZUL 879105 IC50 = 690 nM T11211 C4PK6E 1273173 IC50 = 500 nM T11211 C57NQA 1481979 IC50 = 2260 nM T11211 C26BJU 1490756 IC50 = 1590 nM T11211 CVYN41 1490776 IC50 = 620 nM T11211 C4GAI8 1653625 IC50 > 200000 nM T11211 CYX38L 1713996 IC50 = 1800 nM T11211 COWR13 1736098 IC50 = 4000 nM T11211 CWEV20 1821509 IC50 = 250 nM T11211 CGD23L 1834356 EC50 > 10000 nM T11211 CP3RV7 1834359 EC50 > 10000 nM T11211 C0KNE5 1935870 IC50 = 12000 nM T11211 CB2LE7 1944110 IC50 = 21000 nM T11211 CW61XD 2254186 IC50 = 1900 nM T11211 CB6Z2Q 2258754 IC50 > 200000 nM T11211 CM03LE 2526709 IC50 > 10000 nM T11211 CQ5ZK1 2537506 EC50 = 7300 nM T11211 C3WZ4K 2566134 IC50 = 50000 nM T11211 CJ05TV 2640256 IC50 = 7000 nM T11211 CP30MO 2772455 IC50 = 19000 nM T11211 CWKV50 2772508 IC50 > 200000 nM T11211 CI2S8N 2772636 IC50 = 12000 nM T11211 CZ5C8O 2772641 IC50 = 50000 nM T11211 C9TWA7 2772706 IC50 = 163800 nM T11211 CDA80M 2772715 IC50 > 200000 nM T11211 CTDB12 2772716 IC50 > 200000 nM T11211 C65DER 2772722 IC50 > 200000 nM T11211 C9BU1Y 2772726 IC50 > 200000 nM T11211 CKN4V8 2788122 IC50 = 5090 nM T11211 CD6L8G 2808235 IC50 = 26240 nM T11211 CFXU19 2857621 IC50 > 200000 nM T11211 C3KP5M 2863715 IC50 = 8200 nM T11211 C9O0IE 2865710 IC50 = 36840 nM T11211 C2UW1R 2885298 IC50 = 5000 nM T11211 CTBC06 2941086 EC50 > 10000 nM T11211 CQXE70 2952744 EC50 > 10000 nM T11211 C2EHS5 2952945 EC50 > 10000 nM T11211 CRK2I6 3114779 IC50 = 13100 nM T11211 C0CUX1 3160911 EC50 > 10000 nM T11211 CPM30Q 3435316 IC50 = 22 nM T11211 CMW5A9 4430623 EC50 = 41 nM T11211 CX5W6P 4529791 IC50 > 200000 nM T11211 C9-MAY-08 4531195 IC50 = 9840 nM T11211 CW71VC 5106787 IC50 = 2730 nM T11211 CQ78BW 5287785 Ki = 0.3 nM T11211 C9C0OW 5288215 Ki = 6.1 nM T11211 CQIC09 5377516 IC50 = 1510 nM T11211 C2OX9F 5387866 IC50 = 5920 nM T11211 C46CXW 5709142 IC50 = 3500 nM T11211 CCPM14 5709228 IC50 = 5250 nM T11211 C3G6IQ 5736172 IC50 > 10000 nM T11211 C83TPI 5736234 IC50 < 1000 nM T11211 C3XHT9 6035059 IC50 = 5010 nM T11211 CEZF05 6092405 IC50 = 5950 nM T11211 C4Z1FT 6161872 IC50 = 4360 nM T11211 C1I7GF 6211950 IC50 < 1000 nM T11211 C16ZSG 6439929 IC50 = 220 nM T11211 CE7C2H 6625430 IC50 = 7410 nM T11211 C96CJY 6876440 IC50 = 17900 nM T11211 CKR60D 7019274 IC50 = 420000 nM T11211 CP8H0Q 7256489 IC50 = 400 nM T11211 CP45AI 7529104 IC50 = 3910 nM T11211 CAE6J4 8326955 IC50 = 62000 nM T11211 C3XZS2 8910877 EC50 > 25000 nM T11211 CRM32Y 9796274 Ki = 11 nM T11211 C8L3JO 9798904 IC50 = 72 nM T11211 CY2DK5 9799659 IC50 = 503 nM T11211 C7REX1 9805004 IC50 = 630.96 nM T11211 C0PBZ7 9817592 IC50 = 725 nM T11211 CZ5O8I 9817655 IC50 = 42 nM T11211 C3K2BP 9817717 Ki = 33 nM T11211 CT73GV 9817870 IC50 > 1000 nM T11211 CQ4KC5 9818071 IC50 = 244 nM T11211 C8LGV3 9818136 Ki = 16 nM T11211 C4TJ8E 9818221 EC50 = 2.4 nM T11211 CRF9I3 9818222 Ki = 96 nM T11211 CL68PO 9820051 EC50 = 0.4 nM T11211 C8A3WG 9820510 EC50 = 7.8 nM T11211 CAS62V 9820859 IC50 = 72 nM T11211 C06RXB 9821393 Ki = 2660 nM T11211 C45TEL 9821984 IC50 = 889 nM T11211 C87QGC 9822077 EC50 = 77 nM T11211 C7HGB0 9822150 IC50 = 820 nM T11211 CBU0D4 9822809 EC50 = 3.2 nM T11211 CD9S5P 9825465 Ki = 3115 nM T11211 CY7M9S 9838735 IC50 = 22 nM T11211 CE62WD 9839013 IC50 = 210 nM T11211 CBS8M2 9839134 IC50 = 1292 nM T11211 C8HZ6B 9839661 EC50 = 26 nM T11211 C6J1GC 9839747 Ki = 4.2 nM T11211 C1JEL7 9841234 IC50 = 467 nM T11211 C92CPK 9841404 EC50 = 3.5 nM T11211 CK7UC3 9841413 EC50 = 2.3 nM T11211 C0BA9I 9841791 IC50 = 17 nM T11211 C6MDS5 9842220 Ki > 1000 nM T11211 C7P6XH 9842832 EC50 = 6 nM T11211 C17HVF 9843571 EC50 = 5.9 nM T11211 C96ENK 9844232 EC50 = 22 nM T11211 C9R6FO 9844328 EC50 = 27 nM T11211 CBL0G7 9845028 EC50 = 5.9 nM T11211 C7N6XE 9846167 EC50 = 2.3 nM T11211 C7RS9U 9846657 Ki > 5000 nM T11211 CERF28 9861044 Ki = 1.2 nM T11211 C96HIZ 9861667 IC50 = 30 nM T11211 C3K4EU 9862027 EC50 = 14 nM T11211 C26AVW 9862171 IC50 = 30 nM T11211 CW3QG6 9862271 IC50 = 251 nM T11211 C7HYF1 9863591 IC50 = 479 nM T11211 C7J4BX 9864637 EC50 = 2.7 nM T11211 CKMP85 9864638 EC50 = 15 nM T11211 CMY5I9 9865500 EC50 = 2 nM T11211 CR90XE 9866074 EC50 = 1.6 nM T11211 CVP2K0 9869358 IC50 = 1300 nM T11211 C7DU4F 9879175 Ki = 14.9 nM T11211 C01ZFV 9882789 IC50 > 10000 nM T11211 CXR1H8 9882950 IC50 = 9 nM T11211 C2B8AX 9884451 Ki = 20 nM T11211 CHSD36 9884851 EC50 = 0.9 nM T11211 CEM27C 9885473 IC50 = 650 nM T11211 C0IJM9 9885493 EC50 = 3.8 nM T11211 CTR69M 9885897 EC50 = 0.2 nM T11211 C4QYU8 9888073 Ki > 1000 nM T11211 C85LEV 9888362 IC50 = 34 nM T11211 CKDT60 9889057 IC50 = 660 nM T11211 CZ5R9B 9890023 Ki = 3360 nM T11211 C9K2DW 9890426 IC50 = 190 nM T11211 CG5HV9 9903918 Ki = 113 nM T11211 C2M7HE 9904204 IC50 = 1.4 nM T11211 CJ7U3R 9904286 EC50 = 2 nM T11211 C39AXH 9904328 EC50 = 2.2 nM T11211 C6SWK1 9904610 IC50 = 207 nM T11211 CO85QN 9904758 IC50 = 31 nM T11211 CTI1J8 9905296 EC50 = 1.4 nM T11211 C2PW1X 9905402 EC50 = 3.2 nM T11211 CI7XD1 9905853 EC50 = 1.9 nM T11211 CE1TK2 9908041 IC50 = 795 nM T11211 CIS37A 9908086 Ki = 96 nM T11211 CC39QB 9908246 IC50 = 785 nM T11211 CI2Q9D 9915554 IC50 = 350 nM T11211 CMJG42 9921530 IC50 = 129 nM T11211 C1D4SN 9921561 IC50 = 1500 nM T11211 C91TNX 9925682 Ki = 5 nM T11211 CU5WR0 9925752 IC50 = 25 nM T11211 C8SAF2 9926254 IC50 = 27 nM T11211 CADN52 9927250 Ki = 9 nM T11211 C53YWQ 9927342 EC50 = 3.9 nM T11211 CG06MI 9927792 EC50 = 0.4 nM T11211 CQ68ZH 9929654 IC50 = 5.5 nM T11211 CUK3E9 9933829 EC50 > 2500 nM T11211 C24FUO 9943699 IC50 = 280 nM T11211 CC5Z8A 9948080 Ki > 1000 nM T11211 CZVR83 9948117 Ki = 26 nM T11211 C8FK6G 9948118 EC50 = 13 nM T11211 C0YVS2 9948631 Ki = 1.7 nM T11211 CC6X7Q 9948659 EC50 = 52 nM T11211 CAJ69U 9949233 Ki > 1000 nM T11211 C95VKG 9949253 IC50 = 751 nM T11211 CCSX75 9949772 IC50 = 377 nM T11211 C6P3AO 9949959 IC50 = 675 nM T11211 C8NP5S 9951041 Ki = 0.9 nM T11211 CIT48E 9951393 EC50 = 0.5 nM T11211 CKU64T 9952569 IC50 > 10000 nM T11211 C4TM1W 9952803 EC50 = 27 nM T11211 CW0ED9 9953456 IC50 = 180 nM T11211 C1P7QW 9953889 EC50 = 2 nM T11211 CVW2A7 9954090 EC50 = 4.2 nM T11211 CMQ31W 9955467 IC50 = 636 nM T11211 CJV68Y 9967148 Ki = 1.5 nM T11211 C95CAN 9978625 Ki = 9.74 nM T11211 CP2E8A 9979395 IC50 = 238 nM T11211 C1QP8T 9993897 EC50 = 5 nM T11211 C4V6RF 9998996 IC50 > 5000 nM T11211 C52ADB 10023861 Ki = 560 nM T11211 CNE3X9 10025526 IC50 > 10000 nM T11211 CQ9GX5 10025527 IC50 = 170 nM T11211 CJBQ93 10067789 Ki = 16.5 nM T11211 CFY67M 10070808 IC50 = 315 nM T11211 CBD2T3 10088392 EC50 = 0.3 nM T11211 CM3OR5 10125985 IC50 = 45 nM T11211 CD9EV1 10126599 EC50 = 62 nM T11211 C1WYS8 10127169 EC50 = 8 nM T11211 CQM6E2 10149720 EC50 = 119 nM T11211 CPV5Z4 10149838 IC50 = 100 nM T11211 CR6N7C 10156793 Ki = 96.3 nM T11211 C0MX7K 10157532 IC50 > 10000 nM T11211 CSHY89 10172243 IC50 = 24 nM T11211 CQ6JH8 10173083 EC50 = 8 nM T11211 C8L7HJ 10179031 IC50 > 10000 nM T11211 CLJ02H 10194468 EC50 = 14 nM T11211 CV0LE4 10194889 IC50 > 1000 nM T11211 CH52XQ 10199298 IC50 = 296 nM T11211 C3LPF6 10199303 IC50 = 16.5 nM T11211 CKE61Q 10220715 IC50 = 34 nM T11211 CD1H2S 10221453 Ki = 15 nM T11211 CJ9BE0 10222329 IC50 > 10000 nM T11211 C84SRT 10223610 IC50 > 10000 nM T11211 C18FMW 10237542 EC50 = 138 nM T11211 CQGN38 10237827 EC50 = 12 nM T11211 C1WO5H 10250179 IC50 = 340 nM T11211 CLP9J3 10260561 IC50 = 90 nM T11211 CH9CJ8 10269417 EC50 = 190 nM T11211 CR59SC 10271193 IC50 = 6525 nM T11211 CPIS57 10271557 IC50 > 10000 nM T11211 C5S6GI 10287404 IC50 = 292 nM T11211 CUQC81 10287415 EC50 = 17 nM T11211 C8FMU2 10294401 EC50 = 3.5 nM T11211 CLJU03 10298892 Ki = 3066 nM T11211 CB9YD2 10308517 IC50 = 180 nM T11211 C1W5ZD 10308681 EC50 = 17 nM T11211 C3M1VR 10309552 EC50 = 26 nM T11211 C9FCQ5 10313926 IC50 = 60 nM T11211 CX7WS4 10316069 IC50 = 745 nM T11211 CJB8R4 10319017 Ki = 1177 nM T11211 CEB82Z 10337245 Ki = 1099 nM T11211 CQP1Y7 10340204 IC50 = 1550 nM T11211 CZ05VX 10355755 IC50 = 1621.81 nM T11211 CIL31A 10358742 Ki = 2 nM T11211 CDBZ06 10372181 IC50 = 1600 nM T11211 C6RQK1 10386584 IC50 > 10000 nM T11211 C59VXD 10386752 IC50 > 4000 nM T11211 CZ5CJ3 10423330 IC50 = 250 nM T11211 C37VXR 10432143 IC50 = 449 nM T11211 C1KE6C 10446402 IC50 = 494 nM T11211 CVW6O0 10448918 Ki = 16 nM T11211 C0NT9D 10454007 IC50 > 5000 nM T11211 C1H5RP 10458842 EC50 > 10000 nM T11211 CO84SF 10470625 EC50 = 9 nM T11211 CYQ65Z 10472575 IC50 = 0.009 nM T11211 CUL8O4 10475384 IC50 > 5000 nM T11211 C8O1QG 10476314 Ki = 698 nM T11211 CYE7C2 10496255 Ki = 1644 nM T11211 CT7IG5 10497270 Ki = 1139 nM T11211 CO35TR 10499308 Ki = 6810 nM T11211 C5N7PW 10500864 IC50 = 23000 nM T11211 C6FA1N 10501542 Ki = 3008 nM T11211 C5AP6C 10503520 IC50 = 1236 nM T11211 C5WP1Q 10517398 Ki = 6454 nM T11211 C63ENM 10518992 IC50 = 26 nM T11211 CB0RC3 10520975 IC50 = 57 nM T11211 CR1OS9 10523126 Ki = 1075 nM T11211 C5CDF0 10524606 Ki = 6387 nM T11211 CYS8J9 10546095 Ki 10000 nM T11211 C7R9MN 10552375 Ki = 1.65 nM T11211 CRKM07 10564291 IC50 < 1000 nM T11211 CZ31QX 10567979 Ki = 17 nM T11211 C96GWO 10567980 IC50 = 42 nM T11211 C87UQF 10568861 Ki = 874 nM T11211 CCOE17 10591908 IC50 = 34 nM T11211 CB04AE 10593144 Ki = 1542 nM T11211 CBEC38 10596252 IC50 = 1220 nM T11211 C6G7JR 10596379 Ki = 620 nM T11211 CC8T7J 10598305 IC50 = 946 nM T11211 CGQK63 10610968 IC50 = 36 nM T11211 CEI98J 10614884 IC50 = 23 nM T11211 C3W1BN 10615956 IC50 = 27 nM T11211 CBJ8N5 10615957 IC50 = 27 nM T11211 CXUS14 10615958 Ki = 46 nM T11211 C47WCB 10617171 Ki = 80.9 nM T11211 CAD6L2 10618033 Ki = 696 nM T11211 CO3V0S 10622594 IC50 = 481 nM T11211 C1U0KY 10640594 Ki = 39 nM T11211 C57PFY 10643931 Ki = 504 nM T11211 C02ZMG 10643956 IC50 = 253 nM T11211 CF08PC 10661117 Ki > 10000 nM T11211 C97HTI 10662571 IC50 = 28 nM T11211 C1RIM7 10662717 IC50 = 30 nM T11211 C3RTS7 10663608 IC50 = 23 nM T11211 CU9X3A 10665612 Ki = 1449 nM T11211 C69CNF 10667548 Ki = 1196 nM T11211 CYNG45 10668755 Ki = 887 nM T11211 CS6YF0 10690456 Ki = 732 nM T11211 CYRQ10 10691647 Ki = 1400 nM T11211 C6SP3O 10694256 Ki = 1091 nM T11211 CY81CQ 10710954 IC50 = 156 nM T11211 C1Q0BO 10710955 Ki = 169 nM T11211 CP7G8A 10711095 IC50 = 22 nM T11211 CVD2Y9 10717098 IC50 = 1089 nM T11211 CK2NM9 10717832 Ki = 807 nM T11211 CIU2Q7 10733732 IC50 = 36 nM T11211 CG3MQ7 10734760 IC50 = 48 nM T11211 C1MA4E 10735732 IC50 = 159 nM T11211 CUG2Z9 10739308 Ki = 1942 nM T11211 CAT1X8 10741366 IC50 = 401 nM T11211 C3H6CZ 10754393 Ki > 10000 nM T11211 CBHG38 10758309 Ki = 151 nM T11211 CRF6B3 10759291 IC50 = 27 nM T11211 CB3JD0 10763832 Ki = 1457 nM T11211 CJ4D6M 10782071 IC50 = 68 nM T11211 CEC5Z2 10782232 IC50 = 164 nM T11211 C7HAB1 10782276 Ki = 1923 nM T11211 CNV27D 10783127 Ki = 1518 nM T11211 C7EF4Q 10783200 Ki = 10 nM T11211 CNL1U7 10785305 Ki = 6662 nM T11211 C07BOR 10787258 IC50 = 1426 nM T11211 C10AMX 10805958 Ki = 570 nM T11211 C35YZT 10806774 Ki = 9 nM T11211 CBX48C 10807828 Ki = 1591 nM T11211 CN5WV4 10809583 Ki = 2318 nM T11211 C1CRQ5 10811045 IC50 = 916 nM T11211 CL7JN6 10827013 Ki = 2698 nM T11211 C4NWT7 10829815 IC50 = 46 nM T11211 CD4G1K 10830667 Ki = 670 nM T11211 CN1H5Z 10832792 IC50 = 1239 nM T11211 CYRE47 10851308 IC50 = 27 nM T11211 CP4K9Q 10853414 IC50 = 83 nM T11211 CX68SV 10854490 IC50 = 31 nM T11211 CA96PR 10860931 Ki = 2590 nM T11211 CHU9A4 10873317 Ki = 1589 nM T11211 CI5F0S 10881662 Ki > 1000 nM T11211 CK41RM 10892050 Ki > 10000 nM T11211 CBD12K 10906044 Ki = 819 nM T11211 C2UG0A 10937849 IC50 = 640 nM T11211 C5GJ3U 10956165 IC50 = 330 nM T11211 CHU10G 10960295 Ki = 960 nM T11211 CT2BR8 10969959 Ki = 239 nM T11211 C07JFA 10993685 Ki > 1000 nM T11211 CUC05J 11002535 Ki = 1320 nM T11211 C7E9XI 11015162 Ki = 439 nM T11211 CRH3L8 11025398 IC50 = 900 nM T11211 CU02DM 11046701 Ki = 2460 nM T11211 CIH8K4 11066740 Ki = 1300 nM T11211 CI8GJ5 11079263 IC50 = 258 nM T11211 C09ZLY 11088436 Ki = 54 nM T11211 C6T7CR 11089159 Ki > 5000 nM T11211 C6LYG7 11090322 IC50 = 250 nM T11211 C6BN3Y 11098040 IC50 = 363.08 nM T11211 CE2O8Y 11110616 Ki = 650 nM T11211 C1OJK3 11131414 Ki = 2060 nM T11211 CXS6J7 11155441 Ki = 150 nM T11211 CJ7KZ9 11155655 Ki = 4.6 nM T11211 CU4ME5 11162285 IC50 = 6 nM T11211 CO07NW 11179835 IC50 = 49 nM T11211 CS2P7O 11185187 IC50 = 0.8 nM T11211 CVAI71 11186162 IC50 = 1768 nM T11211 CJGR94 11204416 IC50 > 1000 nM T11211 C4U0DF 11213029 Ki = 290 nM T11211 CW7GQ2 11220011 Ki = 2.2 nM T11211 CI13LE 11220450 Ki = 1.9 nM T11211 CLCM91 11224044 Ki = 570 nM T11211 CRN4V2 11232136 IC50 > 3000 nM T11211 C27QRB 11236228 IC50 = 110 nM T11211 C0H9VJ 11247872 IC50 = 30 nM T11211 CNJ4Q3 11255230 IC50 > 5000 nM T11211 C4S3EI 11276892 IC50 = 7 nM T11211 CC0XI4 11279959 IC50 = 325 nM T11211 C4SC0W 11281576 IC50 > 5000 nM T11211 CUX0S2 11282904 Ki = 290 nM T11211 CKIH41 11301122 Ki = 0.5 nM T11211 CN3ER0 11304696 IC50 = 79 nM T11211 C0XUF2 11305564 IC50 > 5000 nM T11211 C68HGD 11308236 IC50 = 346 nM T11211 CUB9T4 11311771 IC50 = 78 nM T11211 CT9Y4O 11339440 IC50 = 775 nM T11211 CP2DL0 11377050 IC50 = 3600 nM T11211 C98VQF 11382272 Ki = 0.45 nM T11211 CI5Q3B 11384987 IC50 = 160 nM T11211 C70LDA 11394286 Ki = 2.3 nM T11211 C8B9VO 11397073 IC50 = 3700 nM T11211 CPH2O3 11399042 IC50 = 332 nM T11211 CU7IE0 11410199 IC50 = 11700 nM T11211 CO20QH 11416730 IC50 = 215 nM T11211 CA8SF7 11426706 IC50 = 123 nM T11211 CC9D7U 11427021 IC50 = 1717 nM T11211 CTE02B 11428355 Ki = 0.3 nM T11211 CH3DA9 11428356 Ki = 0.3 nM T11211 C5WO0U 11429662 IC50 > 5000 nM T11211 COAZ62 11444005 IC50 = 77 nM T11211 CC75NQ 11477616 Ki = 630 nM T11211 CF2LU7 11482282 IC50 = 3.8 nM T11211 CQ62KS 11485693 IC50 = 690 nM T11211 C1I9YX 11493141 IC50 = 42 nM T11211 C9Q1NY 11494167 Ki = 780 nM T11211 CU20CR 11507567 IC50 = 2.11 nM T11211 CM2RQ4 11518267 IC50 = 470 nM T11211 C1G5KI 11525374 Ki = 1508 nM T11211 CY85BV 11529436 IC50 = 72 nM T11211 C61NXQ 11532117 IC50 = 1200 nM T11211 C5E8BW 11532211 IC50 = 730 nM T11211 C9G5AE 11536973 IC50 = 169 nM T11211 C5W8HY 11537063 IC50 = 11 nM T11211 C2OK8A 11539440 IC50 = 7800 nM T11211 CBDT68 11539442 IC50 = 120 nM T11211 CMSQ72 11539737 IC50 = 250 nM T11211 C7SNY2 11551147 IC50 = 1000 nM T11211 CR4D8K 11558528 IC50 = 33 nM T11211 CL6FW4 11564970 IC50 > 10000 nM T11211 C19NWZ 11565922 IC50 = 718 nM T11211 C3YOM0 11566011 IC50 = 216 nM T11211 CB37YF 11566981 Ki = 50 nM T11211 C2FEY6 11568732 Ki = 1170 nM T11211 CUX53M 11573689 Ki = 44 nM T11211 CZ10OF 11575288 IC50 = 680 nM T11211 CK7WN9 11575794 IC50 = 140 nM T11211 CY9BI7 11580582 IC50 = 257 nM T11211 CKC76H 11589004 IC50 = 51 nM T11211 CQI75K 11594758 IC50 = 42 nM T11211 CZ54QN 11594953 IC50 = 157 nM T11211 C7FVU1 11602515 IC50 = 430 nM T11211 C7YS3I 11609033 IC50 = 60 nM T11211 C0NB5I 11611466 IC50 > 10000 nM T11211 C4JBS6 11616298 IC50 = 354 nM T11211 CSB97O 11617028 Ki = 57 nM T11211 CLN5X6 11618173 IC50 = 1900 nM T11211 C5CHR7 11623463 IC50 = 127 nM T11211 C6LRT7 11623735 IC50 = 22 nM T11211 CB10RY 11623915 IC50 = 85 nM T11211 CZY25E 11624290 Ki = 29 nM T11211 C7K5DW 11630910 IC50 = 69 nM T11211 C8M6GX 11631082 IC50 = 843 nM T11211 C0RD7O 11633120 IC50 > 10000 nM T11211 CF98ZL 11633474 IC50 = 100 nM T11211 CQG0J3 11638442 EC50 = 0.2512 nM T11211 C60DQS 11638602 IC50 = 1436 nM T11211 C6AFP7 11639214 IC50 > 5000 nM T11211 C7NBT6 11645733 IC50 = 172 nM T11211 COES01 11646102 Ki = 8.2 nM T11211 CPY64Q 11652455 IC50 = 120 nM T11211 C8V6ER 11652714 IC50 = 545 nM T11211 C2QTU1 11655725 IC50 = 100 nM T11211 C7R5AC 11659526 IC50 = 103 nM T11211 CZ8IJ6 11659900 Ki = 189 nM T11211 CHKJ71 11661370 IC50 = 4600 nM T11211 C74SAZ 11661683 IC50 = 370 nM T11211 C7O8RH 11662271 IC50 = 500 nM T11211 C0LEZ3 11667800 Ki = 915 nM T11211 CR28PS 11667973 IC50 = 37 nM T11211 C49OHB 11668856 IC50 = 130 nM T11211 CEC7P6 11673811 IC50 = 60 nM T11211 C3VE2O 11675775 IC50 > 10000 nM T11211 CJL8A6 11681415 IC50 = 287 nM T11211 CO15VB 11689938 IC50 = 1000 nM T11211 C4KG8V 11690220 IC50 = 330 nM T11211 CPWR20 11690589 IC50 = 170 nM T11211 C5I9KT 11695011 IC50 = 13 nM T11211 CXR9Z7 11695104 IC50 = 113 nM T11211 C02BAO 11695574 Ki = 14 nM T11211 CQ73SI 11697622 IC50 = 200 nM T11211 CBA95Q 11697749 IC50 = 440 nM T11211 CEU9G7 11698066 IC50 = 1100 nM T11211 C2OPH3 11698067 IC50 > 5000 nM T11211 C1AVI5 11698085 IC50 = 220 nM T11211 CC6VK8 11702683 IC50 = 3767 nM T11211 CVUM48 11710191 Ki = 36 nM T11211 C9CUP1 11715539 EC50 = 2.5 nM T11211 C8QI2G 11719005 IC50 = 190 nM T11211 CR52IJ 11722356 IC50 = 7.9 nM T11211 C4OH1Y 11726899 Ki = 690 nM T11211 CZ0B7H 11731863 IC50 = 215 nM T11211 C4DCI8 11738269 IC50 = 33 nM T11211 CR12UX 11738282 IC50 = 20 nM T11211 C9I3LZ 11738605 IC50 = 718 nM T11211 CV49MT 11747706 IC50 = 0.2 nM T11211 CY1F4I 11752649 Ki = 1900 nM T11211 C9VA5N 11779973 IC50 = 11100 nM T11211 CR70FP 11794088 Ki = 1497 nM T11211 CU7EJ1 11822858 Ki = 180 nM T11211 C6VM0J 12002222 IC50 = 32 nM T11211 C2LY7R 12002243 IC50 = 24 nM T11211 C4U8KY 12085089 IC50 = 8727 nM T11211 C4TRW3 12112694 IC50 = 336 nM T11211 CT1Q6A 12317197 IC50 > 10000 nM T11211 CN6OL5 12439548 IC50 = 7510 nM T11211 C86INA 12607025 IC50 > 200000 nM T11211 C3X5KO 12713141 IC50 = 50 nM T11211 C2HZR1 13145095 IC50 = 8690 nM T11211 C0J1XB 13440714 IC50 = 890 nM T11211 CY6TJ2 14596455 IC50 = 2960 nM T11211 C3DW2I 15308132 IC50 = 460 nM T11211 CB7Q3A 15440425 Ki = 18 nM T11211 C14LTD 15463551 IC50 > 1000 nM T11211 CSJ9W0 15517884 Ki = 29 nM T11211 CB7K0N 15521393 IC50 = 4500 nM T11211 C96KXP 15521394 IC50 > 10000 nM T11211 CRW4K7 15521395 IC50 > 10000 nM T11211 C3F1KG 15952779 IC50 = 100 nM T11211 C69GUF 15959081 IC50 = 860 nM T11211 C8YCP1 16016075 IC50 > 200000 nM T11211 CMZH47 16051364 IC50 = 100 nM T11211 CE8F4N 16090309 EC50 = 2.1 nM T11211 CFZ54L 16090310 EC50 = 1.5 nM T11211 C5RZ2V 16090311 Ki = 222 nM T11211 CX4O6F 16090312 EC50 = 1.9 nM T11211 C39HMG 16090313 EC50 = 2.8 nM T11211 CC24LB 16110489 EC50 > 10000 nM T11211 CO1J7K 16124540 IC50 = 11 nM T11211 C1Q5SV 16220168 IC50 = 3600 nM T11211 CQL72W 16539500 IC50 = 5000 nM T11211 CTDR16 16626366 IC50 = 32900 nM T11211 C7O0EH 16645516 IC50 = 28560 nM T11211 C8UT4N 16658899 Ki = 206 nM T11211 CH6CN0 16658901 EC50 = 2.7 nM T11211 CCF69R 16658902 Ki = 19 nM T11211 CY91RP 16659398 EC50 = 31 nM T11211 C1UY8J 16666386 IC50 > 1000 nM T11211 CWK35C 16730429 IC50 = 7700 nM T11211 C0N5KD 16731512 Ki = 1.6 nM T11211 CJM8B3 16731514 Ki = 2.9 nM T11211 C4Y1PJ 16731515 Ki = 0.7 nM T11211 C31QVA 16731844 Ki = 1.9 nM T11211 C8V9ZU 16731845 EC50 = 2.1 nM T11211 CU0LA8 16731847 Ki = 23 nM T11211 C07YFR 16731998 Ki = 4 nM T11211 C9BC0L 16732000 Ki = 0.9 nM T11211 CG7V8Y 16732137 Ki = 2.3 nM T11211 C68GWF 16732139 Ki = 0.9 nM T11211 C75TYX 16732140 Ki = 1 nM T11211 C5IGM3 16733585 Ki = 2 nM T11211 CGW48S 16733766 Ki = 1.5 nM T11211 CEB3D8 16769319 IC50 = 5040 nM T11211 CW82LP 17027902 IC50 > 200000 nM T11211 C4F6KI 17027949 IC50 > 200000 nM T11211 C82LQX 17027986 IC50 > 200000 nM T11211 CWVG01 17027987 IC50 = 40300 nM T11211 CY4T1I 17027988 IC50 = 30600 nM T11211 C2SVJ9 17028005 IC50 = 12700 nM T11211 CG9M0J 17028006 IC50 = 11100 nM T11211 CGC74M 17028025 IC50 > 200000 nM T11211 CW6LU7 17028045 IC50 = 24100 nM T11211 CMI90S 17028047 IC50 = 45000 nM T11211 CV1O8I 17028048 IC50 = 13700 nM T11211 CEG87D 17028050 IC50 > 200000 nM T11211 CP6D0S 17144586 EC50 = 20300 nM T11211 C82RKN 17399143 IC50 = 1380 nM T11211 CSKX58 17758233 Ki = 1530 nM T11211 C7CPW9 17758234 Ki = 110 nM T11211 CI5KT6 17758236 Ki = 346 nM T11211 C3FP7L 17921933 IC50 = 1248 nM T11211 CWJ06U 18106212 EC50 = 12600 nM T11211 C0C5HO 18111026 EC50 = 14500 nM T11211 CX03YG 18188955 IC50 > 10000 nM T11211 CR19ST 18512166 IC50 = 170 nM T11211 CEN14G 18512334 IC50 = 300 nM T11211 CBI64N 18551237 IC50 = 501.19 nM T11211 C30ZFV 18753314 IC50 = 210 nM T11211 CHI5T3 18756402 Ki = 5.5 nM T11211 C03OAG 19133039 IC50 = 29040 nM T11211 C1ZBX7 19566931 IC50 = 600 nM T11211 C95KIE 20160413 IC50 = 25000 nM T11211 C5ZYJ0 20231824 Ki = 355 nM T11211 C7KC2V 20587845 EC50 = 2.6 nM T11211 C50ZMW 20587865 Ki = 43 nM T11211 CEH7V5 20786216 IC50 > 1000 nM T11211 CB40FM 21094319 EC50 = 410 nM T11211 C6VEB4 21094321 EC50 > 10000 nM T11211 C5HO9W 21094361 EC50 = 394 nM T11211 CL9WF6 21176636 IC50 = 13670 nM T11211 CF0S6J 21210483 IC50 = 5300 nM T11211 C97WCO 21941658 IC50 = 158.49 nM T11211 CCI89R 21948853 IC50 > 1000 nM T11211 CB2SF4 21948904 IC50 > 1000 nM T11211 C2ZP7V 22218142 EC50 = 9 nM T11211 CU30DZ 22252955 Ki = 3.5 nM T11211 CF0K2J 22278979 Ki = 36 nM T11211 CHPY76 22278998 IC50 = 504 nM T11211 CT9M4C 22279012 IC50 = 30 nM T11211 CA7Y0I 22279020 Ki = 110 nM T11211 C3TC9X 22279031 IC50 = 56 nM T11211 C3GUJ1 22279035 IC50 = 98 nM T11211 CE6X4S 22279036 Ki = 9 nM T11211 CMC62X 22279038 IC50 = 149 nM T11211 CTP1U5 22279049 IC50 = 301 nM T11211 COF0D8 22279076 Ki = 5.4 nM T11211 CSO14A 22279116 Ki = 15 nM T11211 C42MYX 22279130 Ki = 13 nM T11211 C5T4WQ 22279141 Ki = 50 nM T11211 C7IW0K 22279155 Ki = 157 nM T11211 C1KFV4 22279178 IC50 = 2 nM T11211 C42QLS 22279187 Ki = 30 nM T11211 CXGM37 22279207 Ki = 118 nM T11211 C8RA7S 22279210 Ki = 163 nM T11211 CS57PT 22279252 Ki = 761 nM T11211 C04YEG 22279256 IC50 = 507 nM T11211 CC68FS 22279268 Ki = 20 nM T11211 CUL15Y 22279277 Ki = 641 nM T11211 CPS5T1 22279290 Ki = 29 nM T11211 C8Z7ES 22279296 EC50 = 0.8 nM T11211 C02DTL 22279311 IC50 = 32 nM T11211 CTJS03 22279315 IC50 = 43 nM T11211 C10MNP 22279323 Ki = 65 nM T11211 CDK02G 23030191 IC50 = 47 nM T11211 C1ZET4 23030294 IC50 = 310 nM T11211 C7WS8G 23030352 IC50 = 6.7 nM T11211 CK4L3U 23079916 EC50 = 21 nM T11211 C6UZD7 23433503 IC50 = 1460 nM T11211 CGY94Z 23433542 IC50 = 1110 nM T11211 C84MWR 23433579 IC50 = 788 nM T11211 C9O6RB 23596322 Ki > 10000 nM T11211 C2NVK3 23598977 Ki = 24 nM T11211 CPG1L3 23598979 Ki = 1 nM T11211 CG07ZK 23613735 IC50 = 35000 nM T11211 CONM26 23613737 IC50 = 14100 nM T11211 C8HFZ5 23613764 IC50 > 200000 nM T11211 CGB28T 23631256 EC50 = 21 nM T11211 CX8VB7 23631257 Ki = 10 nM T11211 CBQ01G 23631259 Ki = 7.6 nM T11211 CI85NX 23644730 Ki = 24 nM T11211 CX7A6L 23647974 EC50 = 7.8 nM T11211 CZ25GU 23648042 Ki = 11 nM T11211 CCZ08D 23648043 Ki = 463 nM T11211 CAHI31 23648044 Ki = 30 nM T11211 CK6A4D 23648045 Ki = 241 nM T11211 CU7S5A 23648046 EC50 = 73 nM T11211 CN2DP9 23648047 IC50 = 111 nM T11211 C46VKA 23648048 EC50 = 0.4 nM T11211 C34ZVB 23648049 EC50 = 1.3 nM T11211 CG46VA 23648050 EC50 = 6.8 nM T11211 C8AM1P 23648051 EC50 = 1.8 nM T11211 CW2F8C 23648052 EC50 = 81 nM T11211 C0ERI3 23648053 EC50 = 5.9 nM T11211 CK1C4N 23648054 EC50 = 46 nM T11211 CHND27 23648055 Ki = 6.6 nM T11211 CC3AK5 23648056 EC50 = 12 nM T11211 CCU54F 23648057 Ki = 19 nM T11211 CT27QS 23648060 IC50 = 36 nM T11211 CV87PS 23648061 Ki = 0.4 nM T11211 C49CAO 23648062 Ki = 0.5 nM T11211 C7JM4Z 23648063 Ki = 0.5 nM T11211 CQ5HO0 23648064 Ki = 23 nM T11211 CY0P5A 23648066 EC50 = 2.3 nM T11211 C4HO3J 23648067 IC50 = 20 nM T11211 CA2QD8 23648068 EC50 = 3.7 nM T11211 CI92LB 23648069 EC50 = 3.6 nM T11211 CS2ZV3 23648070 EC50 = 3.2 nM T11211 CM6NZ9 23648214 IC50 > 10000 nM T11211 C7TX5D 23729483 IC50 = 7 nM T11211 C2YK6I 23847279 IC50 = 520 nM T11211 CWPH96 24180508 IC50 = 1000 nM T11211 CZ9N1A 24180647 IC50 = 39.9 nM T11211 CZI4C6 24739672 Ki = 1740 nM T11211 CS23KY 24739834 Ki = 490 nM T11211 C1M9QG 24739836 Ki = 2590 nM T11211 CG5SJ0 24739997 Ki > 3900 nM T11211 C7Z1HW 24740156 Ki = 2550 nM T11211 CTE1N2 24748569 EC50 > 10000 nM T11211 C4WYE7 24749678 Ki = 849 nM T11211 CY2JS4 24749684 Ki = 676 nM T11211 C2QHO3 24749808 Ki = 211 nM T11211 C5SIN1 24752898 Ki = 12 nM T11211 C5S6JN 24780149 IC50 > 1000 nM T11211 CW5TJ7 24781731 IC50 > 1000 nM T11211 CIT41F 24784464 IC50 = 320 nM T11211 C8F7WP 24811980 IC50 = 9.6 nM T11211 CNM45B 24850992 EC50 = 1 nM T11211 C1JTW2 24851053 Ki = 5.98 nM T11211 CC53XL 24860583 Ki > 2300 nM T11211 C9RLM8 24865155 IC50 = 2.9 nM T11211 C58NZJ 24865524 Ki = 45 nM T11211 CGE0V4 24882669 IC50 > 10000 nM T11211 C58RHY 24883011 IC50 > 10000 nM T11211 CW35CK 24883012 IC50 > 10000 nM T11211 C3SC0V 24883054 IC50 > 10000 nM T11211 C4SA6C 24883055 IC50 > 10000 nM T11211 C9E0ZK 24892822 Ki = 1.7 nM T11211 C5LZK2 24895096 EC50 = 1800 nM T11211 C2PGW1 24896626 IC50 = 560 nM T11211 C97QRS 24936209 Ki = 1000 nM T11211 COGP96 24936313 Ki > 5000 nM T11211 CVY09S 24936449 Ki > 5000 nM T11211 CBN24H 24936982 Ki = 2513 nM T11211 C06PDG 24952192 Ki = 2341 nM T11211 CG1CF9 24952193 Ki = 696 nM T11211 CZC7L8 24953162 IC50 > 5000 nM T11211 C4W7BN 24954947 IC50 > 5000 nM T11211 C6XC2R 24954951 IC50 > 10000 nM T11211 C5XGK8 24986664 EC50 = 0.29 nM T11211 C0LIQ3 24987377 IC50 = 100 nM T11211 CHY0D7 25013322 IC50 > 5000 nM T11211 C0TPS5 25013653 IC50 > 10000 nM T11211 CWU91M 25013811 IC50 > 20000 nM T11211 CSH29L 25013812 IC50 > 10000 nM T11211 CQAW47 25016975 IC50 = 27 nM T11211 CI50YU 25016977 IC50 = 0.8 nM T11211 CVMQ72 25016978 EC50 = 208 nM T11211 CAW0R1 25017238 IC50 = 112 nM T11211 C76TPO 25017239 IC50 = 62 nM T11211 C5MY3D 25017241 EC50 = 50 nM T11211 CLEH69 25017242 IC50 = 144 nM T11211 C6GWE8 25017244 IC50 = 0.3 nM T11211 C9EZX1 25017509 IC50 = 1.1 nM T11211 CC0E9P 25017511 Ki = 4 nM T11211 CNCX17 25017513 Ki = 5 nM T11211 C1N0WL 25017760 Ki = 21 nM T11211 C1NGB9 25017761 EC50 = 18 nM T11211 CYW0N8 25017765 Ki = 3 nM T11211 CYLC08 25017766 Ki = 50 nM T11211 C25EFU 25018011 Ki = 27 nM T11211 CXH61M 25018012 Ki = 8 nM T11211 C2G1JK 25053351 Ki > 30000 nM T11211 CAW8M0 25070694 IC50 = 740 nM T11211 CWJ38T 25093228 IC50 > 3000 nM T11211 CWUA34 25093229 IC50 = 26 nM T11211 C80QXO 25093230 IC50 = 1599 nM T11211 C9Z1YD 25129860 Ki = 1500 nM T11211 CK9A5R 25132127 IC50 = 400 nM T11211 C58LFZ 25141236 Ki = 5 nM T11211 C35HKY 25145080 Ki = 490 nM T11211 CXF9G0 25145082 Ki = 110 nM T11211 C21XDY 25145083 Ki = 96 nM T11211 CANT87 25145217 Ki = 39 nM T11211 CE1I7A 25145499 Ki = 1214 nM T11211 CV6N1P 25145500 Ki = 64 nM T11211 CS6JQ1 25167502 Ki = 1500 nM T11211 C2TJ3P 25191004 IC50 = 6000 nM T11211 C98JQI 25218466 IC50 > 10000 nM T11211 CR8F9X 25218467 IC50 > 10000 nM T11211 C87ARD 25225237 IC50 = 50000 nM T11211 CLY9W3 25235364 IC50 > 10000 nM T11211 CLO1F8 25236617 EC50 = 14400 nM T11211 CKUP63 25236633 EC50 > 25000 nM T11211 C3FW0Y 25257459 IC50 > 10000 nM T11211 CY6X2V 25258136 IC50 = 420 nM T11211 CV4Y6N 25258138 IC50 > 10000 nM T11211 CLX0P9 25258381 IC50 = 880 nM T11211 CNLS64 25258386 IC50 > 10000 nM T11211 C5G4VI 25764492 IC50 = 1200 nM T11211 COX54F 25808053 IC50 = 900 nM T11211 C8AP2Q 32408099 IC50 = 6470 nM T11211 CB0D1T 34282649 EC50 > 25000 nM T11211 C5OKE6 35875974 EC50 > 25000 nM T11211 C4GSR9 35901875 IC50 = 1513.56 nM T11211 CU2B0C 36925618 EC50 = 15200 nM T11211 CCTW62 36925632 EC50 = 1700 nM T11211 CU3N1T 42618084 Ki = 0.8 nM T11211 CWC96V 42618085 Ki = 0.3 nM T11211 CF76VY 42618086 Ki = 0.2 nM T11211 CQ70JS 42618088 Ki = 10 nM T11211 CFD79C 42618089 Ki = 19 nM T11211 CG0E4V 42635876 IC50 = 234.42 nM T11211 C4UWJ5 43138564 IC50 = 123 nM T11211 C4H3YS 43138588 IC50 = 315 nM T11211 C8BGR0 43320715 IC50 = 10 nM T11211 CSY8D9 43320717 IC50 > 10000 nM T11211 C1JE8M 43320720 IC50 = 6650 nM T11211 C4K6TQ 43320726 IC50 = 2720 nM T11211 C4W9CM 43320729 IC50 > 10000 nM T11211 CR4C2X 43320749 IC50 = 54 nM T11211 CQP8E7 43364282 IC50 = 20 nM T11211 CD61KH 44125830 IC50 = 10715.19 nM T11211 CPB8S3 44125832 IC50 = 3715.35 nM T11211 CX89HM 44138106 Ki = 2900 nM T11211 CCJ3S4 44222256 EC50 = 26 nM T11211 CE0U8G 44222257 EC50 = 2 nM T11211 CC3XR6 44222258 EC50 = 5 nM T11211 CW1EM8 44222259 IC50 = 715 nM T11211 C8UFH0 44240547 IC50 = 110 nM T11211 C6AO4R 44240549 IC50 = 340 nM T11211 C10XAL 44240606 IC50 = 720 nM T11211 C0OGD2 44240609 IC50 = 190 nM T11211 CQ93RI 44247563 IC50 = 11 nM T11211 C8G4VL 44263921 Ki = 24 nM T11211 CA58OB 44263937 Ki = 7 nM T11211 C27GEW 44263978 Ki = 21 nM T11211 CM1N6W 44263979 Ki = 9 nM T11211 CV48KP 44264011 Ki = 12 nM T11211 C6F2RD 44264068 Ki = 8 nM T11211 CR8U3J 44264069 Ki = 22 nM T11211 C6EQO3 44264273 EC50 = 7 nM T11211 C8GZ1T 44264292 Ki = 6 nM T11211 CG87FY 44264293 IC50 = 24 nM T11211 CQAI15 44264294 Ki = 11 nM T11211 CF5R4O 44264299 IC50 = 42 nM T11211 C9RTV4 44264322 Ki = 109 nM T11211 C71LUI 44264348 Ki = 15 nM T11211 CF8AO1 44264372 EC50 = 10 nM T11211 CJ4UF9 44264412 Ki = 42 nM T11211 CKQA48 44264433 EC50 = 16 nM T11211 CP2LY4 44264458 Ki = 23 nM T11211 CB53OG 44264482 EC50 = 8 nM T11211 C0OA6M 44264483 EC50 = 2 nM T11211 C5LYK2 44264503 IC50 = 7 nM T11211 COCE32 44264569 EC50 = 2 nM T11211 C4XT3H 44264575 IC50 = 5 nM T11211 CH05UD 44264578 EC50 = 209 nM T11211 CXOR54 44264579 EC50 = 5 nM T11211 C01HSQ 44264588 EC50 = 1 nM T11211 CHK23J 44276210 EC50 = 10 nM T11211 C60HMY 44276220 Ki = 58 nM T11211 CE74KN 44276221 Ki = 12 nM T11211 CJHQ43 44276222 IC50 = 251 nM T11211 CM5L0K 44276347 Ki = 22 nM T11211 CM63QL 44276359 EC50 = 19 nM T11211 CAU6Q2 44276415 Ki = 8 nM T11211 C1C7UD 44276534 EC50 = 137 nM T11211 CTF9O7 44276554 Ki = 9 nM T11211 CH6UZ2 44276555 EC50 = 3 nM T11211 C80NPS 44276579 Ki = 2 nM T11211 CH15DK 44276580 EC50 = 7 nM T11211 CO0BA7 44276581 Ki = 8 nM T11211 COM4B6 44276587 EC50 = 158 nM T11211 COKV03 44276600 EC50 = 2 nM T11211 CKAD39 44276822 IC50 = 12 nM T11211 C97GND 44276823 IC50 = 216 nM T11211 C9A5IM 44276824 Ki = 9 nM T11211 CP8OC7 44282950 Ki = 621 nM T11211 C6X2IH 44295653 Ki 10000 nM T11211 C0X9EZ 44295844 Ki = 1.1 nM T11211 C1DBA2 44305237 IC50 = 250 nM T11211 CDB54J 44305270 IC50 > 1000 nM T11211 C0XLN6 44305556 IC50 = 6.1 nM T11211 CHB82F 44305684 IC50 = 395 nM T11211 C1UK4M 44305720 IC50 = 60 nM T11211 CTW67P 44305733 IC50 = 90 nM T11211 CD7C5E 44305809 IC50 = 147 nM T11211 CH4PU5 44305819 IC50 > 10000 nM T11211 CDXK57 44305874 IC50 = 644 nM T11211 C6N1AR 44305929 IC50 = 63 nM T11211 C9U6SZ 44306067 IC50 = 428 nM T11211 CW21CA 44317747 Ki = 90 nM T11211 CT62WI 44341706 Ki = 886 nM T11211 CO10KF 44341745 Ki = 456 nM T11211 CP0AQ3 44341860 Ki = 785 nM T11211 CE62XL 44341871 Ki = 2046 nM T11211 CIFK12 44341872 Ki = 1485 nM T11211 C6KSD0 44341876 Ki = 903 nM T11211 CP6LV3 44341880 Ki = 1330 nM T11211 C8RQS2 44342092 Ki = 697 nM T11211 CDGP02 44353994 IC50 = 203 nM T11211 C73CXK 44354006 Ki > 1000 nM T11211 CJ6F4A 44354487 Ki > 1000 nM T11211 CL5P7M 44354744 Ki > 1000 nM T11211 CN16XG 44354803 IC50 = 45 nM T11211 C0N3TD 44354884 IC50 = 1100 nM T11211 CPQ2A6 44354885 IC50 = 45 nM T11211 CM0G1V 44354886 IC50 = 200 nM T11211 CL6G3Q 44355066 IC50 = 150 nM T11211 CSAU31 44377064 IC50 = 7 nM T11211 CG45XW 44377072 Ki = 63 nM T11211 CPI21A 44377073 Ki = 194 nM T11211 C7H9NC 44377081 Ki = 10 nM T11211 C60DYH 44377090 Ki = 5 nM T11211 CGC91Q 44377091 Ki = 33 nM T11211 CEX2Y0 44377092 Ki = 9 nM T11211 CPNG27 44377093 Ki = 21 nM T11211 CVH2R3 44377098 Ki = 4 nM T11211 CME56K 44377100 IC50 = 54 nM T11211 CYLI63 44377110 IC50 = 48 nM T11211 CI0P8B 44377165 Ki = 167 nM T11211 C7Y3AD 44377166 IC50 = 27 nM T11211 C1GN8P 44377167 IC50 = 26 nM T11211 CLB1C4 44377168 IC50 = 56 nM T11211 CDKG72 44377250 Ki = 10 nM T11211 C5GK9E 44377264 IC50 = 10 nM T11211 CR5H4T 44377266 Ki = 23 nM T11211 C8QSU3 44377274 Ki = 9 nM T11211 CQX39I 44377356 IC50 = 51 nM T11211 C6ZMH3 44377379 Ki = 17 nM T11211 CH6PK8 44377380 IC50 = 53 nM T11211 C10BGN 44377381 Ki = 9 nM T11211 C9FJW4 44377382 Ki = 21 nM T11211 CDJ5F4 44377395 IC50 = 23 nM T11211 C13SYV 44396250 Ki = 17 nM T11211 CB1P0S 44396251 Ki = 4.6 nM T11211 CHY1C3 44396271 Ki = 34 nM T11211 C29MBI 44396272 Ki = 21 nM T11211 C4TQ6N 44396282 Ki = 8.1 nM T11211 CH2Y3L 44396283 Ki = 7.4 nM T11211 CWZB52 44396284 Ki = 16 nM T11211 CD80LM 44396296 Ki = 8.9 nM T11211 C6SI5L 44396297 Ki = 6.2 nM T11211 CR4H1E 44396316 Ki = 34 nM T11211 C45LRH 44396317 Ki = 8.9 nM T11211 C5JG6H 44396330 Ki = 53 nM T11211 CA8V4G 44396331 Ki = 37 nM T11211 C57CPQ 44396332 Ki = 18 nM T11211 CHG9O1 44396490 IC50 = 0.9 nM T11211 CPQL46 44396502 IC50 = 17 nM T11211 CNH4C3 44396512 IC50 = 61 nM T11211 C1OYG3 44396526 IC50 = 0.2 nM T11211 CO25DV 44396547 IC50 = 2 nM T11211 CUT91V 44397094 IC50 = 780 nM T11211 CFVU42 44397206 IC50 = 90 nM T11211 CCE5G7 44397286 Ki = 40 nM T11211 C9TJ8P 44397478 Ki = 240 nM T11211 C8L7HT 44404365 Ki = 3380 nM T11211 CPQV14 44404372 Ki = 2900 nM T11211 C79JEI 44407631 IC50 = 1761 nM T11211 CB0L6S 44407636 IC50 = 3733 nM T11211 C2W0PF 44407655 IC50 > 5000 nM T11211 CWU1O4 44407658 IC50 = 1769 nM T11211 C6J3VA 44407760 IC50 = 1402 nM T11211 C1O6WJ 44407763 IC50 = 4617 nM T11211 C21CBM 44407771 IC50 > 5000 nM T11211 CD3E0R 44407782 IC50 = 20 nM T11211 C2O1DA 44407785 IC50 = 120 nM T11211 CXD31Y 44407857 IC50 = 7.9 nM T11211 CAVO39 44418759 Ki = 1.5 nM T11211 CH1R7M 44420600 EC50 > 10000 nM T11211 CXCG59 44421996 IC50 = 420 nM T11211 CFL86B 44421999 IC50 = 420 nM T11211 C19GYL 44422001 IC50 = 190 nM T11211 CM8I0R 44422004 IC50 = 120 nM T11211 CC46UT 44422008 IC50 = 730 nM T11211 C3A6XY 44422014 IC50 = 300 nM T11211 C3C7LG 44422020 IC50 = 490 nM T11211 C2V8GT 44422030 IC50 = 260 nM T11211 C7DAZ6 44422031 IC50 = 480 nM T11211 C37HWF 44422034 IC50 = 940 nM T11211 C20FOR 44422037 IC50 = 1800 nM T11211 C6HKN3 44422041 IC50 = 6300 nM T11211 CSMB47 44422043 IC50 = 6800 nM T11211 C7ZCY4 44422044 IC50 = 960 nM T11211 CAVQ81 44422045 IC50 = 110 nM T11211 CMN2V0 44422046 IC50 > 10000 nM T11211 C19RLO 44422047 IC50 = 6600 nM T11211 C4Z6MS 44422052 IC50 = 10000 nM T11211 C67DTU 44422053 IC50 = 280 nM T11211 C2R5IW 44422054 IC50 = 110 nM T11211 CLM57N 44422057 IC50 = 550 nM T11211 C0K3NV 44422058 IC50 = 330 nM T11211 CDF95J 44422064 IC50 = 570 nM T11211 CAX3E7 44422065 IC50 = 1300 nM T11211 C3JG9N 44422066 IC50 = 9900 nM T11211 CE2I7N 44422067 IC50 = 820 nM T11211 CT8DI2 44422068 IC50 > 10000 nM T11211 CE8L7N 44422075 IC50 = 280 nM T11211 C84GWS 44422080 IC50 = 300 nM T11211 CGWD03 44432383 Ki = 20 nM T11211 CR3OW8 44433502 IC50 < 1000 nM T11211 C1Z0QH 44433503 IC50 < 1000 nM T11211 C3SJ5V 44433504 Ki = 590 nM T11211 CC6N4M 44433644 IC50 = 410 nM T11211 CVLS95 44433645 IC50 = 350 nM T11211 C9SHW3 44433649 IC50 = 600 nM T11211 C86HYW 44433650 IC50 = 300 nM T11211 CRF74O 44433651 IC50 = 430 nM T11211 C3QMB7 44433653 IC50 = 660 nM T11211 C92BRW 44433654 IC50 = 5800 nM T11211 COWV92 44433655 IC50 = 850 nM T11211 CB8UO0 44433656 IC50 = 96 nM T11211 C3QR6X 44433657 IC50 = 420 nM T11211 C0LVE3 44433659 IC50 = 670 nM T11211 C6VZ3R 44433663 IC50 = 120 nM T11211 CJOS78 44434090 IC50 = 9.8 nM T11211 C3MDG1 44434091 IC50 = 20.1 nM T11211 C58WSK 44434092 IC50 = 140 nM T11211 C0BZA5 44434093 IC50 = 0.8 nM T11211 CX6O9M 44434094 IC50 = 229 nM T11211 CSA20N 44434095 IC50 = 61.2 nM T11211 CNF01X 44434096 IC50 = 146 nM T11211 CQ5T7O 44434097 IC50 = 1900 nM T11211 CATL94 44434098 IC50 = 200 nM T11211 CVU53K 44434100 IC50 = 14.7 nM T11211 CAL4P8 44434102 IC50 = 989 nM T11211 CB9R5M 44434103 IC50 = 1310 nM T11211 C01PME 44434104 IC50 > 10000 nM T11211 CUJ9P1 44434105 IC50 = 2230 nM T11211 C8CGU2 44434106 IC50 = 1540 nM T11211 CK7GQ8 44434108 IC50 = 8140 nM T11211 C3LO1U 44440237 IC50 = 33 nM T11211 CLK05T 44440238 IC50 = 88 nM T11211 CP3JU8 44440239 IC50 = 15 nM T11211 C34ERB 44440240 IC50 = 85 nM T11211 C5KG7L 44440241 IC50 = 68 nM T11211 CB1ZS3 44440262 IC50 = 1375 nM T11211 CKON02 44440263 IC50 = 1120 nM T11211 C5DB8N 44440264 IC50 = 710 nM T11211 C89JEW 44440265 IC50 > 1000 nM T11211 CR7G2K 44440266 IC50 > 1000 nM T11211 CVT4O9 44440267 IC50 > 1000 nM T11211 CO98DZ 44440268 IC50 > 1000 nM T11211 CL3WI5 44441857 IC50 = 842 nM T11211 CIL2C9 44441858 IC50 = 2610 nM T11211 CR2S3A 44441859 IC50 = 500 nM T11211 C6GRK9 44441860 IC50 = 3160 nM T11211 CA1BY2 44441862 IC50 = 520 nM T11211 C6SMB2 44441863 IC50 = 1615 nM T11211 CTQ15A 44441864 IC50 = 170 nM T11211 CF06VH 44441865 IC50 = 290 nM T11211 C1X5MS 44441866 IC50 = 330 nM T11211 C8BI2Z 44442001 IC50 = 209 nM T11211 C92EZP 44442002 IC50 = 136 nM T11211 COP18N 44442003 IC50 = 169 nM T11211 CR96IG 44442004 IC50 = 1700 nM T11211 CPW05D 44442005 IC50 = 4926 nM T11211 CFM0Y1 44442939 EC50 = 5.4 nM T11211 C7JSI6 44442940 IC50 = 72 nM T11211 CXZ5G6 44442945 IC50 = 84 nM T11211 C1OWF9 44442946 IC50 = 1480 nM T11211 C49EKQ 44442947 IC50 = 113 nM T11211 CKG9M6 44442948 EC50 > 10000 nM T11211 C9SV4G 44442949 EC50 = 420 nM T11211 CD69TR 44442950 EC50 = 406 nM T11211 CKO85I 44442952 EC50 = 228 nM T11211 C9A7EN 44442959 EC50 = 51 nM T11211 CVUB54 44442961 EC50 = 227 nM T11211 CK60AI 44442963 EC50 = 300 nM T11211 C6Y2RA 44442966 EC50 = 276 nM T11211 CZCH50 44442968 EC50 = 272 nM T11211 C6B2WZ 44442969 EC50 = 20 nM T11211 C8G4OX 44442970 EC50 = 35 nM T11211 CX3IU4 44442971 EC50 = 43 nM T11211 CYZ5D1 44442973 EC50 = 98 nM T11211 CT5B7F 44442974 IC50 = 65 nM T11211 C60HBZ 44442975 IC50 = 45 nM T11211 CME9N5 44442976 EC50 = 18 nM T11211 CJA9L8 44443100 IC50 = 2 nM T11211 CKI23S 44443116 IC50 = 17 nM T11211 C2O4JQ 44444354 IC50 = 43 nM T11211 C3RV5X 44448568 Ki = 11 nM T11211 CT52FO 44448685 IC50 = 0.2 nM T11211 C5C8XN 44448708 EC50 = 1.1 nM T11211 CJ3I9N 44448709 EC50 = 11 nM T11211 CAOZ50 44448756 EC50 = 1.3 nM T11211 CW16NM 44448784 Ki = 32 nM T11211 C0QV9G 44448787 Ki = 2.6 nM T11211 C1I0JD 44448818 IC50 = 25 nM T11211 C95YNE 44448819 Ki = 18 nM T11211 CQBW46 44448960 EC50 = 6.6 nM T11211 C5G3LU 44448962 EC50 = 11 nM T11211 C51IQO 44449150 IC50 = 44 nM T11211 CBT7A9 44449152 EC50 = 36 nM T11211 C2JE9X 44449183 Ki = 1.1 nM T11211 C5HU8E 44449184 Ki = 180 nM T11211 CW3T6Q 44449185 Ki = 150 nM T11211 CQGB87 44449210 Ki = 1.3 nM T11211 CMT39O 44449211 IC50 = 51 nM T11211 CF4DV9 44449212 Ki = 2.4 nM T11211 CK30BP 44449214 Ki = 18 nM T11211 CYPI98 44454211 Ki = 40 nM T11211 CZ1Y7T 44455867 Ki = 1100 nM T11211 C8I4CF 44455886 Ki = 1000 nM T11211 CBV4A3 44455888 Ki = 1100 nM T11211 CVXA65 44462785 IC50 = 100 nM T11211 CR5SI0 44476535 EC50 > 10000 nM T11211 CAWJ02 44512434 EC50 = 1.585 nM T11211 CGZ64T 44550719 IC50 = 31.7 nM T11211 CF6V4G 44563171 EC50 > 10000 nM T11211 CIR72Y 44564657 IC50 = 35 nM T11211 CL2S8N 44564658 IC50 = 702 nM T11211 CY5SU8 44564660 IC50 = 167 nM T11211 CS6J3Q 44565103 IC50 > 10000 nM T11211 C62FLW 44565203 IC50 = 56 nM T11211 C73FNX 44565204 IC50 = 411 nM T11211 CK8MH3 44565647 Ki > 10000 nM T11211 CMWE31 44568326 Ki = 3100 nM T11211 CB1CO2 44568327 Ki = 4900 nM T11211 C0CLK1 44568328 Ki = 6100 nM T11211 CSP8H4 44568329 Ki = 2700 nM T11211 CB72AX 44568330 Ki = 2700 nM T11211 CP3AK8 44568352 Ki = 490 nM T11211 C5BL1A 44568353 Ki = 350 nM T11211 CW8D4B 44568354 Ki = 690 nM T11211 CU4SH1 44568355 Ki = 2200 nM T11211 C8MFH4 44568356 Ki = 3600 nM T11211 C6OM2E 44568381 Ki = 2000 nM T11211 C9W6LD 44568382 Ki = 3400 nM T11211 C8IC4S 44568383 Ki = 520 nM T11211 CIG4A2 44568384 Ki = 140 nM T11211 CACM15 44568408 Ki = 130 nM T11211 CK8O4P 44568409 Ki = 330 nM T11211 CD59WQ 44568410 IC50 = 13700 nM T11211 CYLE93 44568411 Ki = 1400 nM T11211 CCP5M3 44568457 Ki = 1300 nM T11211 CTV97R 44568458 Ki = 49 nM T11211 CWHP14 44568459 Ki = 6 nM T11211 CV81MH 44568460 Ki = 36 nM T11211 CXLM16 44568496 Ki = 130 nM T11211 C7YU4N 44568497 Ki = 7 nM T11211 C9JFN4 44568498 Ki = 100 nM T11211 C3LA8D 44568499 Ki = 170 nM T11211 C3RVO4 44568500 Ki = 3 nM T11211 C3SNC2 44568540 Ki = 220 nM T11211 CJ5ZR1 44568541 Ki = 3 nM T11211 CR7TS6 44568542 IC50 = 6100 nM T11211 C4L0ES 44568543 Ki = 27 nM T11211 C8X3IJ 44568586 Ki = 9 nM T11211 CQS41M 44568587 Ki = 340 nM T11211 C65GHE 44568588 Ki = 370 nM T11211 CFJ54O 44574243 Ki = 1.1 nM T11211 C8BGL6 44585565 IC50 > 3000 nM T11211 CA1Y5L 44591817 Ki = 0.7 nM T11211 C3KUD4 44591818 Ki = 17 nM T11211 CV9T0G 44592067 IC50 = 202 nM T11211 CFB0L3 44592068 IC50 = 2280 nM T11211 CYL52U 44592099 IC50 = 34 nM T11211 CJ3VI8 44593465 Ki = 9300 nM T11211 CIJP09 44605898 IC50 > 10000 nM T11211 CT5G6Z 45101436 IC50 = 1995.26 nM T11211 C97ZET 45269449 IC50 = 250 nM T11211 C08UBE 45272032 IC50 = 1600 nM T11211 CN3G7M 45272695 EC50 = 5 nM T11211 C57EZH 45275745 IC50 > 10000 nM T11211 C98WDQ 45485494 EC50 > 10000 nM T11211 CB2LO0 45485501 EC50 > 10000 nM T11211 C96THD 45485556 EC50 > 10000 nM T11211 CRP29T 45485557 EC50 > 10000 nM T11211 CR8I9S 45486375 IC50 > 4000 nM T11211 CP35QW 45486376 IC50 > 4000 nM T11211 C4XDQ1 45486377 IC50 > 4000 nM T11211 CDA24N 45486383 IC50 > 4000 nM T11211 C9YM2G 45486384 IC50 > 4000 nM T11211 CX8HO5 45486385 IC50 > 4000 nM T11211 CJX89Y 45486393 IC50 > 4000 nM T11211 C8K2DM 45486403 IC50 > 4000 nM T11211 CQT1C9 45486404 IC50 > 4000 nM T11211 C0RID5 45486424 IC50 > 4000 nM T11211 COG73H 45486437 IC50 > 4000 nM T11211 C2NWO7 45486438 IC50 > 4000 nM T11211 CM8F4H 45486439 IC50 > 4000 nM T11211 CW20GE 45486443 IC50 > 4000 nM T11211 C5HL9V 45486450 IC50 > 4000 nM T11211 CW7J5K 45486451 IC50 > 4000 nM T11211 CL91NK 45486456 IC50 > 4000 nM T11211 C6OYN8 45486457 IC50 > 4000 nM T11211 C3KU7H 45486464 IC50 > 4000 nM T11211 C14DQK 45486465 IC50 > 4000 nM T11211 CR6P7Z 45486470 IC50 > 4000 nM T11211 CU3IY5 45486473 IC50 > 4000 nM T11211 CHRX37 45486474 IC50 > 4000 nM T11211 CY54HC 45486477 IC50 > 4000 nM T11211 CX8LZ0 45486478 IC50 > 4000 nM T11211 C7PMW0 45486484 IC50 > 4000 nM T11211 COD9R1 45486485 IC50 > 4000 nM T11211 CBNI02 46830477 IC50 = 44 nM T11211 C1RJV2 46830478 IC50 = 28 nM T11211 C1BYW8 46830503 IC50 > 10000 nM T11211 C04BWG 46830504 IC50 > 10000 nM T11211 CY2ZJ0 46830505 IC50 > 10000 nM T11211 CC45TP 46830506 IC50 > 10000 nM T11211 CN7Q8A 46830507 IC50 > 10000 nM T11211 C0QT3G 46830795 IC50 > 10000 nM T11211 C0JCX3 46830796 IC50 > 10000 nM T11211 CMS6R9 46830797 IC50 > 10000 nM T11211 CJIN74 46830798 IC50 > 10000 nM T11211 CRY31M 46830799 IC50 > 10000 nM T11211 CKA07I 46830800 IC50 > 10000 nM T11211 C4XRF9 46830801 IC50 > 10000 nM T11211 C2NC3V 46831087 IC50 > 10000 nM T11211 CXP6K3 46831397 IC50 > 10000 nM T11211 C0QNC9 46831400 IC50 > 10000 nM T11211 CX6L7Q 46831696 IC50 = 3162.28 nM T11211 CQ1IP3 46831697 IC50 = 10000 nM T11211 CL1KR4 46831698 IC50 = 6309.57 nM T11211 C1DH9W 46831699 IC50 = 6309.57 nM T11211 CASV14 46831700 IC50 = 5011.87 nM T11211 CTXY26 46831701 IC50 = 5011.87 nM T11211 CG0J5K 46831956 IC50 > 10000 nM T11211 CY3WK4 46831957 IC50 = 3162.28 nM T11211 CP19UN 46831958 IC50 = 6309.57 nM T11211 CBJZ85 46831959 IC50 > 10000 nM T11211 CE4VC8 46831960 IC50 > 10000 nM T11211 CAR23U 46832233 IC50 > 10000 nM T11211 CUAO43 46832234 IC50 > 10000 nM T11211 CM40EP 46832235 IC50 > 10000 nM T11211 CJ32XT 46832236 IC50 > 10000 nM T11211 C81GUN 46832237 IC50 > 10000 nM T11211 CT31AL 46832511 IC50 > 10000 nM T11211 CR15XE 46832512 IC50 > 10000 nM T11211 CW12GM 46832513 IC50 = 3162.28 nM T11211 C0GTK8 46832514 IC50 = 3981.07 nM T11211 C8HO0L 46832515 IC50 = 2511.89 nM T11211 C2S6PL 46834818 IC50 = 38 nM T11211 CV6E8S 46855605 IC50 = 1480 nM T11211 CD04CW 46871871 Ki = 24.2 nM T11211 CXD42C 46871872 Ki = 342 nM T11211 CRW04Q 46872914 IC50 = 251.19 nM T11211 C4BA9X 46872915 IC50 = 850 nM T11211 CLV41O 46872916 IC50 = 1070 nM T11211 C5IK8F 46873259 IC50 = 1240 nM T11211 C9AFG8 46873260 IC50 = 1990 nM T11211 CXH81W 46873366 IC50 = 190 nM T11211 CW7N8B 46873367 IC50 = 360 nM T11211 CNH28Q 46873368 IC50 = 1200 nM T11211 CPG56I 46888204 IC50 = 55 nM T11211 CZYW10 46888205 IC50 = 200 nM T11211 C2FL6C 46888206 IC50 = 89 nM T11211 CX8J4K 46888265 IC50 > 1000 nM T11211 CO6N0D 46888266 IC50 > 1000 nM T11211 C72MUY 46889765 IC50 > 5000 nM T11211 C6DVO1 46889848 IC50 > 10000 nM T11211 CS8XC4 46893453 IC50 = 5888.44 nM T11211 C8T6RN 46906110 Ki = 283 nM T11211 CP04YQ 46906111 Ki = 493 nM T11211 C4RFX9 46906112 Ki > 10000 nM T11211 CCM4H0 46906113 Ki = 1314 nM T11211 C32JOS 46906137 Ki > 10000 nM T11211 C3GP8J 46906138 Ki = 883 nM T11211 CT0QU8 46906139 Ki > 10000 nM T11211 C16CJP 46906140 Ki = 320 nM T11211 CM4H3Y 46906173 Ki = 636 nM T11211 CU9H2X 46906174 Ki > 10000 nM T11211 CQ2PU6 46906175 Ki = 115 nM T11211 C42RPK 46906176 Ki = 37 nM T11211 CZ7OE3 46906177 Ki = 35 nM T11211 CAK8Y1 46906229 Ki = 64 nM T11211 CE1DN6 46906230 Ki = 406 nM T11211 CT57UI 46906231 Ki = 140 nM T11211 C09VDP 46906256 Ki = 74 nM T11211 CAQT54 46906257 Ki > 10000 nM T11211 CV84RA 46906258 Ki > 10000 nM T11211 CKTU08 46906259 Ki = 203 nM T11211 CGW15V 46906285 Ki > 10000 nM T11211 COMC86 46906286 Ki = 322 nM T11211 CF0UH7 46906482 Ki = 10.4 nM T11211 C3RVF1 46906483 Ki = 2.3 nM T11211 CID4F9 46906484 Ki = 4523 nM T11211 CSK01Q 46906501 Ki = 1531 nM T11211 C7ELM3 46906502 Ki = 3178 nM T11211 CRH1T2 46906503 Ki = 65 nM T11211 C81MYC 46906504 Ki = 51 nM T11211 CAS06I 46906529 Ki = 124 nM T11211 C0I5SR 46906530 Ki = 63 nM T11211 C7BVX3 46906531 Ki = 30 nM T11211 C4BM6J 46906561 Ki = 18 nM T11211 CEP63J 46906562 Ki = 417 nM T11211 CJ9EN0 46906563 Ki = 1010 nM T11211 C3Q7RI 46913890 IC50 > 10000 nM T11211 CP91XE 46914741 IC50 > 10000 nM T11211 CTM2J5 46915203 IC50 > 8920 nM T11211 C75IFZ 46915353 IC50 > 10000 nM T11211 CX70GY 46915355 IC50 > 10000 nM T11211 C7NC4B 46917090 IC50 > 10000 nM T11211 CTVY61 46929339 IC50 = 6200 nM T11211 CL7P3N 46938234 IC50 > 10000 nM T11211 COS28G 46938235 IC50 > 10000 nM T11211 CFJT93 46938236 IC50 = 9050 nM T11211 CHL70M 46938239 IC50 = 9940 nM T11211 C6XKP2 47049885 IC50 = 3320 nM T11211 CW6T1H 49821197 IC50 = 27 nM T11211 CU3S6H 49836028 Ki = 1034 nM T11211 C96SLW 49851364 Ki = 1058 nM T11211 CDN4K6 49851369 Ki = 370 nM T11211 C0K7OD 49851464 Ki > 3000 nM T11211 C4YXN1 49851467 Ki = 993 nM T11211 CI0MX2 49851469 Ki > 4000 nM T11211 CUD91T 49862248 EC50 > 10000 nM T11211 C1NV8O 49862937 Ki = 3.5 nM T11211 C2NE6M 49863247 IC50 = 7.4 nM T11211 CTKV39 49864176 IC50 > 10000 nM T11211 C1G9NP 50925481 IC50 = 13 nM T11211 CZ8J1V 50942115 Ki = 900 nM T11211 CX1KO8 51346768 Ki = 648 nM T11211 C7N9TD 51346823 Ki = 1430 nM T11211 C7U6EA 52941233 IC50 = 500 nM T11211 C03CQM 52941337 IC50 = 95 nM T11211 C7BO9F 52941376 IC50 > 1000 nM T11211 C2ST8Y 52942225 IC50 = 1420 nM T11211 CDP50X 52942229 IC50 = 90 nM T11211 CDV90J 52942528 IC50 > 1000 nM T11211 CUL57E 52943430 IC50 = 34 nM T11211 CAN2T4 52943635 IC50 = 3000 nM T11211 CM8QY5 52943641 IC50 = 80 nM T11211 CNK4V8 52943651 IC50 = 30 nM T11211 CS17IL 52943808 IC50 = 480 nM T11211 CU9OH6 52944606 Ki = 1100 nM T11211 C8Y9SU 52944898 IC50 > 1000 nM T11211 C8GO7A 52945001 IC50 = 34 nM T11211 CQW2E4 52945095 IC50 = 100 nM T11211 C0HZP5 52945868 IC50 = 4600 nM T11211 CUC26Q 52945869 IC50 = 85 nM T11211 CS0X7U 52946488 IC50 = 600 nM T11211 CIC94R 52947094 IC50 = 15 nM T11211 CR4WA9 52947473 IC50 > 10000 nM T11211 CM3VI6 52947474 IC50 = 9200 nM T11211 CD8W0E 52947546 IC50 > 10000 nM T11211 COMY87 52948291 IC50 = 2000 nM T11211 CA1NE7 52948299 IC50 = 34 nM T11211 CQI7C9 52948491 IC50 = 100 nM T11211 CU2CY5 52948638 IC50 > 1000 nM T11211 C06CIL 52949572 Ki = 1800 nM T11211 C7VNH1 52949592 IC50 = 2000 nM T11211 C8K9BT 52949762 IC50 = 50 nM T11211 CK5UT4 53317489 Ki = 403 nM T11211 CM0LU1 53318659 Ki = 400 nM T11211 CUD48O 53320087 Ki = 220 nM T11211 CYH3V0 53325642 Ki = 68.9 nM T11211 C82DYI 53326614 Ki > 4020 nM T11211 CJCP75 53359074 Ki > 5000 nM T11211 CY0AK4 53634112 EC50 = 5 nM T11211 CUR24K 53875787 EC50 = 7 nM T11211 CF6L2Y 54585068 Ki = 2000 nM T11211 C8X5VS 54587024 Ki = 2000 nM T11211 CU9Y7W 54587025 Ki = 2000 nM T11211 C30XLO 54592009 IC50 > 10000 nM T11211 CAN48X 54713170 IC50 = 400 nM T11211 C1IJ8D 54714338 IC50 = 7 nM T11211 CGLX41 55023552 IC50 > 200000 nM T11211 CP17GT 55355450 IC50 = 1460 nM T11211 CCJ42Y 56589543 IC50 = 10000 nM T11211 CR4U9K 56594613 IC50 = 9700 nM T11211 C9ZSC5 56643472 IC50 = 59 nM T11211 CBOE01 56643473 IC50 = 144 nM T11211 CSO36F 56648237 IC50 = 175 nM T11211 CFY6W7 56648316 IC50 = 32 nM T11211 CQ0T1U 56648317 IC50 = 70 nM T11211 CU4RI5 56648318 IC50 = 126 nM T11211 CQ6M7D 56648319 IC50 = 161 nM T11211 C80UYZ 56648320 IC50 = 519 nM T11211 C3JH7S 56648321 IC50 = 82 nM T11211 CDNT13 56648322 IC50 = 75 nM T11211 CSN1A5 56648411 IC50 = 42 nM T11211 C8I3OC 56648412 IC50 = 20 nM T11211 CS53HG 56648413 IC50 = 54 nM T11211 C4LH1V 56648414 IC50 = 30 nM T11211 CMCK31 56648415 IC50 = 16 nM T11211 C75VZD 56648416 IC50 = 69 nM T11211 CV7D0J 56648507 IC50 = 136 nM T11211 CZ84ME 56648508 IC50 = 136 nM T11211 C5H2GD 56648509 IC50 = 90 nM T11211 C02UAS 56648510 IC50 = 163 nM T11211 C4OKC1 56648511 IC50 = 174 nM T11211 CT24OM 56649280 Ki = 68 nM T11211 CXBV25 56659958 IC50 = 399 nM T11211 C87ZYQ 56659959 IC50 = 200 nM T11211 C72XYT 56659964 IC50 = 48 nM T11211 CJV5X7 56659965 IC50 = 43 nM T11211 CZVB12 56663423 IC50 = 10 nM T11211 CNL0W6 56663424 IC50 = 2450 nM T11211 CX08LA 56663425 IC50 = 4910 nM T11211 CR2F0C 56666848 IC50 = 1210 nM T11211 C34SJD 56666849 IC50 = 268 nM T11211 CTJH01 56666852 IC50 = 110 nM T11211 COQ6V5 56666853 IC50 = 28 nM T11211 CJY58N 56666854 IC50 = 215 nM T11211 CV2ZL9 56666855 IC50 = 40 nM T11211 CS3C6I 56670277 IC50 = 2790 nM T11211 CWN86P 56670278 IC50 = 516 nM T11211 CT16GS 56670283 IC50 = 166 nM T11211 C7VL6W 56670284 IC50 = 324 nM T11211 C45STW 56673793 IC50 = 284 nM T11211 C7Z4QK 56673794 IC50 = 17 nM T11211 CRF21W 56673795 IC50 = 17 nM T11211 CSQT70 56677125 IC50 = 766 nM T11211 C3CV8Y 56677130 IC50 = 298 nM T11211 CMH9L6 56677131 IC50 = 174 nM T11211 C3KQ5N 56677132 IC50 = 11 nM T11211 C8AX6T 56677133 IC50 = 880 nM T11211 CU1EO4 56677134 IC50 = 54 nM T11211 C4WFT0 56680439 IC50 = 303 nM T11211 CS8NY4 56680440 IC50 = 3520 nM T11211 CG65LB 56680442 IC50 = 767 nM T11211 CRF32A 56680443 IC50 = 128 nM T11211 CEX6A0 56683767 IC50 = 444 nM T11211 CCY38N 56683768 IC50 = 802 nM T11211 C4X7FR 56683769 IC50 = 1770 nM T11211 CWLZ60 56683770 IC50 = 523 nM T11211 CABE41 56683773 IC50 = 144 nM T11211 CZ20VW 56834944 IC50 = 131 nM T11211 CQ12KI 56837418 IC50 = 40 nM T11211 CF3G2M 56925477 IC50 = 95 nM T11211 CZ7O8G 56925478 IC50 = 1200 nM T11211 CW87RG 56925573 IC50 > 10000 nM T11211 C30DAL 56925669 IC50 = 5900 nM T11211 CQHA65 56925670 IC50 = 4700 nM T11211 CJP31U 56925671 IC50 > 10000 nM T11211 CI3S6F 56925790 IC50 > 10000 nM T11211 CTY1Q9 56925791 IC50 > 10000 nM T11211 CTG9I7 56926011 IC50 = 4500 nM T11211 CJ6D4N 57390869 IC50 = 550 nM T11211 CR63UH 57390870 IC50 = 130 nM T11211 CY0VN5 57390871 IC50 = 120 nM T11211 C1S5TO 57391350 IC50 = 91 nM T11211 CS4Y0Z 57391351 IC50 = 180 nM T11211 CZE53T 57391352 IC50 = 700 nM T11211 C6HRB1 57391422 IC50 = 1200 nM T11211 CBSH29 57391794 IC50 = 266 nM T11211 C5W2CX 57391795 IC50 = 633 nM T11211 C0W9KB 57391796 IC50 = 77 nM T11211 CK4QJ1 57392686 IC50 = 390 nM T11211 C5EKI3 57392687 IC50 = 3.9 nM T11211 CW3L5I 57393119 IC50 = 140 nM T11211 CM4IU9 57394910 IC50 = 160 nM T11211 CW7DJ2 57396151 IC50 = 1500 nM T11211 CG96JP 57396617 IC50 = 510 nM T11211 CZ9V5T 57396618 IC50 = 27 nM T11211 C0HAC5 57397037 IC50 = 105 nM T11211 C54GOD 57398385 IC50 = 0.47 nM T11211 CWK9F0 57398386 IC50 = 110 nM T11211 CZ2MO7 57398435 IC50 = 6300 nM T11211 C24ENR 57398596 IC50 = 68 nM T11211 CO24VD 57398771 IC50 = 71 nM T11211 CLVQ35 57398772 IC50 = 263 nM T11211 C24YLG 57399054 Ki > 5000 nM T11211 CT4U6E 57399615 IC50 = 6500 nM T11211 CZRT27 57400047 IC50 = 53 nM T11211 CHG87W 57400048 IC50 = 26 nM T11211 CCW56F 57400259 IC50 = 337 nM T11211 CAK75B 57400260 IC50 = 977 nM T11211 C0TBY4 57400261 IC50 = 371 nM T11211 CH4M3C 57400425 IC50 = 4100 nM T11211 CJG6M5 57401372 IC50 = 1300 nM T11211 CP26GS 57401373 IC50 = 14 nM T11211 CQY9O0 57401374 IC50 = 78 nM T11211 CF83VM 57401459 Ki > 5000 nM T11211 CC25EM 57401853 IC50 = 180 nM T11211 C8O3KC 57401854 EC50 = 62 nM T11211 C4V2QS 57401855 IC50 = 820 nM T11211 C42FMH 57402062 IC50 = 761 nM T11211 CZK58C 57403124 IC50 = 5 nM T11211 CXTF50 57403125 IC50 = 660 nM T11211 CP68OH 57403565 IC50 = 4200 nM T11211 C6BW2Y 57403630 IC50 = 1600 nM T11211 CK4G0N 57404505 IC50 = 79.6 nM T11211 CX9P8K 57563344 EC50 = 0.15 nM T11211 C3WG0L 57666312 Ki = 700 nM T11211 C43GDR 57666397 Ki = 910 nM T11211 CTM6K5 57690900 IC50 > 1000 nM T11211 C1KZT3 57906156 IC50 > 10000 nM T11211 CQWA53 57926646 IC50 = 1.4 nM T11211 CV3G1D 57926845 IC50 = 1500 nM T11211 CT1EM3 58064710 IC50 > 10000 nM T11211 C8S3EQ 58064714 IC50 = 3250 nM T11211 CPI62D 58064720 IC50 > 10000 nM T11211 CL42XF 58064726 IC50 = 7780 nM T11211 CPL9A6 58064729 IC50 > 10000 nM T11211 CRFS78 58064730 IC50 = 8520 nM T11211 CN1J3V 58064734 IC50 > 10000 nM T11211 CA0SH5 58064735 IC50 > 10000 nM T11211 CI7BP4 58064741 IC50 > 10000 nM T11211 C2FZA7 58064756 IC50 > 10000 nM T11211 CI6XF5 58742295 IC50 = 300 nM T11211 C0JL7A 58973277 IC50 > 1000 nM T11211 C31KUT 59149763 IC50 = 323.59 nM T11211 CH41MU 59149828 IC50 = 1047.13 nM T11211 C2A9JO 59251119 Ki > 5000 nM T11211 CL1TR6 59273014 IC50 = 0.32 nM T11211 C9RI6K 59273018 IC50 = 0.2 nM T11211 CD8A6P 59281281 IC50 = 3700 nM T11211 CBZ0M5 59281312 IC50 > 10000 nM T11211 CCT59B 59281329 IC50 > 10000 nM T11211 CQI5C4 59281343 IC50 > 10000 nM T11211 CPE83R 59281354 IC50 > 10000 nM T11211 CI9EP1 59281363 IC50 > 10000 nM T11211 CQ2BO1 59281403 IC50 > 10000 nM T11211 CP78RD 59281411 IC50 > 10000 nM T11211 CCNU12 59281412 IC50 = 9200 nM T11211 C7HVB1 59281416 IC50 > 10000 nM T11211 CE5A0V 59281447 IC50 > 10000 nM T11211 CZT9S6 59281449 IC50 > 10000 nM T11211 CIKQ89 59281508 IC50 > 10000 nM T11211 CE1A7J 59281531 IC50 > 10000 nM T11211 CK9JZ4 59281538 IC50 > 10000 nM T11211 C4TG5U 59281540 IC50 = 3600 nM T11211 CPC80S 59281541 IC50 = 5600 nM T11211 CXS5C4 59281543 IC50 > 10000 nM T11211 C7KPR9 59281566 IC50 > 10000 nM T11211 CUJP64 59281599 IC50 > 10000 nM T11211 CE8Y1C 59370500 EC50 = 0.19 nM T11211 C8S7UJ 59556904 IC50 = 14 nM T11211 CIFU52 59556909 EC50 = 24 nM T11211 C2P6DK 59556915 EC50 = 1 nM T11211 C4F7OX 59556937 IC50 = 3.4 nM T11211 CUZ1K9 59556948 IC50 = 1.1 nM T11211 CZ2A1X 59556953 EC50 = 3.6 nM T11211 C3IDG5 59556967 IC50 = 9 nM T11211 CH0P4U 59556969 EC50 = 810 nM T11211 CYZI85 59556974 IC50 = 3.6 nM T11211 C6RV5Y 59556985 IC50 = 3.9 nM T11211 C6H8AL 59556999 EC50 = 220 nM T11211 CTY71E 59557018 EC50 = 0.39 nM T11211 CI7W8H 59557020 EC50 = 150 nM T11211 C0AVO7 59557024 EC50 = 1000 nM T11211 C5C3AO 59770003 Ki = 418 nM T11211 C1L4JR 60165333 IC50 = 43 nM T11211 CC4IH9 60195171 IC50 = 446.68 nM T11211 C60AEL 60195172 IC50 = 269.15 nM T11211 C8F9EG 60195173 IC50 = 1479.11 nM T11211 C13IZH 60195174 IC50 = 27.54 nM T11211 CB4JX0 60195175 IC50 = 120.23 nM T11211 C9X4FN 60195176 IC50 = 1096.48 nM T11211 CS85VE 60195262 IC50 = 43.65 nM T11211 CX9M8B 60195263 IC50 = 104.71 nM T11211 CESN14 60195264 IC50 = 10964.78 nM T11211 CA5W6C 60195265 IC50 = 295.12 nM T11211 CAY82V 60195266 IC50 = 707.95 nM T11211 C7C8NQ 60195267 IC50 = 223.87 nM T11211 C8OQR0 60195361 IC50 = 302 nM T11211 CK7I2L 60195362 IC50 = 128.82 nM T11211 CSZR14 60195363 IC50 = 309.03 nM T11211 C03ODG 60195551 IC50 = 616.6 nM T11211 C3MAC6 60195552 IC50 = 2511.89 nM T11211 CTB4D2 60195627 IC50 = 263.03 nM T11211 CAV1N5 60195718 IC50 = 389.05 nM T11211 CC1YT8 60471678 IC50 = 610 nM T11211 C4OD8K 62945565 EC50 = 4700 nM T11211 C0S7VZ 65485745 IC50 = 66 nM T11211 CXY23T 66897267 IC50 = 220 nM T11211 CI1SZ4 66897828 IC50 = 9590 nM T11211 C1CXY9 66996546 IC50 > 10000 nM T11211 CO70AV 67105434 IC50 = 6600 nM T11211 C2NEB3 67339181 IC50 = 1584.89 nM T11211 CL6Y2K 68290392 IC50 = 2940 nM T11211 CW8E0C 68707154 EC50 = 21 nM T11211 CK1F5V 68707555 EC50 = 0.24 nM T11211 C6V1TO 68707868 EC50 = 0.19 nM T11211 C9A6MJ 68709035 EC50 = 2.2 nM T11211 C7MT8P 68709882 EC50 = 0.32 nM T11211 CS3M5E 68710983 EC50 = 0.25 nM T11211 CKPJ76 68711746 EC50 = 2 nM T11211 CN3HP4 68712596 EC50 = 1.2 nM T11211 CV4PD0 68713946 EC50 = 160 nM T11211 CNS26W 68714176 IC50 = 20 nM T11211 CO72WV 69265349 Ki = 28 nM T11211 CB4G2M 69267419 Ki = 8 nM T11211 C5AV1J 69267698 Ki = 3 nM T11211 CE1BP0 69268220 Ki = 3 nM T11211 CO8UN9 69268382 Ki = 3 nM T11211 C3D5GE 69268956 Ki = 3 nM T11211 CU86TA 69269074 Ki = 2 nM T11211 CQTJ47 69269362 Ki = 3 nM T11211 C2OC5M 69790334 IC50 = 1.4 nM T11211 CGR7I3 69802707 IC50 = 34 nM T11211 CF4N1D 70680990 IC50 = 60.6 nM T11211 C80EZU 70680991 IC50 = 301 nM T11211 CXU8R0 70682951 Ki = 4.3 nM T11211 C8QSM2 70683115 IC50 = 170 nM T11211 CJL07F 70683117 IC50 = 197 nM T11211 CARO49 70685018 Ki = 3.3 nM T11211 CW18ZM 70685189 IC50 = 292 nM T11211 C4V9PD 70685190 IC50 = 165 nM T11211 C7CO4X 70689404 IC50 = 126 nM T11211 C61GAS 70691512 IC50 = 293 nM T11211 C4U6HV 70691513 IC50 = 389 nM T11211 CEAG63 70691514 IC50 = 178 nM T11211 CD9M2I 70693604 IC50 = 373 nM T11211 C97DAV 70693605 IC50 = 588 nM T11211 C5QPC0 70697572 Ki = 4.8 nM T11211 CN19MQ 70806890 IC50 = 10500 nM T11211 CIE6Z1 70806946 IC50 = 9540 nM T11211 CR91DC 70960697 IC50 = 68 nM T11211 CX9OH5 70960699 IC50 = 68 nM T11211 CY01GF 70960700 IC50 = 32 nM T11211 C5HM8D 70960701 IC50 = 25 nM T11211 CAOB13 70960753 IC50 = 17 nM T11211 C54SOB 70960760 IC50 = 290 nM T11211 CF8X4I 70960783 IC50 = 370 nM T11211 CI20EO 70960796 IC50 = 1100 nM T11211 C49NKB 71239142 EC50 = 0.4 nM T11211 C9FQ3T 71239150 EC50 = 1.4 nM T11211 CHBZ46 71239205 EC50 = 0.16 nM T11211 CYS31C 71239207 EC50 = 1 nM T11211 C0MX7C 71239311 EC50 = 0.3 nM T11211 CC86FT 71239406 EC50 = 4.5 nM T11211 C7MJQ2 71239416 EC50 = 9.7 nM T11211 CUH71V 71239417 EC50 = 0.5 nM T11211 CP2XF7 71239426 EC50 = 0.93 nM T11211 C2TMQ4 71239443 EC50 = 26 nM T11211 CE9D8Z 71239453 EC50 = 1.5 nM T11211 C7IME2 71239455 EC50 = 7.1 nM T11211 CO6A0N 71244858 EC50 = 978 nM T11211 CV75QC 71449128 EC50 = 56 nM T11211 CH83OP 71449648 IC50 = 977.24 nM T11211 C0FOS8 71451461 IC50 = 2818.38 nM T11211 C94FCP 71452686 IC50 = 0.3 nM T11211 CS1YT8 71452738 IC50 = 63 nM T11211 CH06QW 71453284 IC50 = 1148.15 nM T11211 C7UXM9 71454496 IC50 = 332 nM T11211 C0U5ZF 71455003 IC50 = 13182.57 nM T11211 COH1C0 71456199 EC50 = 16 nM T11211 CU3SE1 71456244 IC50 = 49 nM T11211 CST0R7 71456785 IC50 = 1000 nM T11211 CH76SM 71456786 IC50 = 660.69 nM T11211 CMKD01 71456787 IC50 = 645.65 nM T11211 CZ97CR 71456788 IC50 = 741.31 nM T11211 C53QLH 71456789 IC50 = 79.43 nM T11211 CF08ME 71457470 Ki = 1170 nM T11211 C21BFE 71458005 IC50 = 15 nM T11211 CQA9P7 71459946 EC50 = 7 nM T11211 CEO5G4 71461616 EC50 = 5 nM T11211 C90NUM 71461651 IC50 = 77 nM T11211 CC67FV 71462182 IC50 = 1348.96 nM T11211 C1MHC0 71467246 IC50 = 2800 nM T11211 C4B0IC 71467248 IC50 = 2400 nM T11211 C9JBH6 71508200 IC50 = 27 nM T11211 CNMD32 71508201 IC50 = 1600 nM T11211 CDUM73 71508202 IC50 = 120 nM T11211 C17QCL 71508255 IC50 = 400 nM T11211 CYW34A 71519686 IC50 = 3000 nM T11211 CV8X3O 71541767 IC50 = 9760 nM T11211 C1M6XO 71542719 IC50 = 6260 nM T11211 C0O3RU 71542978 IC50 = 13190 nM T11211 C4E2KX 71542979 IC50 = 5070 nM T11211 CGK4S8 71543393 EC50 = 0.499 nM T11211 C83YJF 71544946 IC50 > 5000 nM T11211 CT9Y5D 71549558 IC50 = 3100 nM T11211 C8ZX0F 71549573 EC50 > 20000 nM T11211 CZ8Y7O 71549829 IC50 = 7700 nM T11211 CPFL57 71549843 IC50 = 12000 nM T11211 CY8SP0 71549969 IC50 = 11000 nM T11211 CX6JR5 71550242 IC50 = 3700 nM T11211 C6WIA2 71550244 IC50 = 3100 nM T11211 CSHT69 71550657 IC50 > 5000 nM T11211 CZ9NW2 71550681 EC50 = 13700 nM T11211 CPN8U4 71550737 EC50 = 0.1 nM T11211 CXZI06 71562914 IC50 > 200000 nM T11211 CYXO53 71582840 IC50 = 1500 nM T11211 C5UM2G 71583169 IC50 > 10000 nM T11211 CLZ6O9 71583170 IC50 > 10000 nM T11211 CX24YH 71583171 IC50 > 10000 nM T11211 CC08YH 71583283 IC50 > 10000 nM T11211 C7MN9Q 71583284 IC50 = 4000 nM T11211 CKS36Y 71583285 IC50 > 10000 nM T11211 C8KGH2 71583287 IC50 = 5800 nM T11211 CDS9K0 71583396 IC50 = 8300 nM T11211 CMC6A8 71583397 IC50 = 6700 nM T11211 CA6T2V 71583398 IC50 = 7400 nM T11211 C37GSP 71681247 IC50 = 2650 nM T11211 CNRU01 71712304 IC50 = 5400 nM T11211 CV39ME 71712305 IC50 = 8200 nM T11211 CWV0E4 71717631 IC50 = 6800 nM T11211 CRFH87 71717693 IC50 = 1000 nM T11211 CU5IZ0 71717985 IC50 > 200000 nM T11211 CZL47I 71717986 IC50 = 55000 nM T11211 C5MA4V 71717987 IC50 > 200000 nM T11211 C0X8SD 71719211 IC50 > 200000 nM T11211 C7AE5H 71719212 IC50 > 200000 nM T11211 CLHZ38 71719213 IC50 = 22800 nM T11211 C02FQE 71719561 IC50 = 2089.3 nM T11211 CMV06D 71719823 IC50 = 5400 nM T11211 C7NO8V 71720428 IC50 > 200000 nM T11211 CQ2DT0 71720429 IC50 > 200000 nM T11211 CNY96D 71730162 IC50 > 10000 nM T11211 C47DEK 71732110 IC50 = 1300 nM T11211 C8OBF3 71732111 IC50 > 10000 nM T11211 C8VC5N 71902847 IC50 = 8430 nM T11211 CP5KM8 72163477 IC50 > 10000 nM T11211 CA6O4K 72163478 IC50 > 10000 nM T11211 C27XWS 72163479 IC50 > 10000 nM T11211 C6M9CN 72163480 IC50 > 10000 nM T11211 CL8AH4 72163481 IC50 > 10000 nM T11211 CB2SD9 72163621 IC50 > 10000 nM T11211 CU6NA8 72163622 IC50 > 10000 nM T11211 CTEV75 72163623 IC50 > 10000 nM T11211 CER73F 72163624 IC50 > 10000 nM T11211 CC8VM7 72163625 IC50 > 10000 nM T11211 CS69AC 72163626 IC50 > 10000 nM T11211 CAJ0H5 72163627 IC50 > 10000 nM T11211 C1D3EU 72163754 IC50 > 10000 nM T11211 C1G3ES 72163755 IC50 > 10000 nM T11211 CP8AC2 72188914 Ki > 25000 nM T11211 CA6FO5 72188915 Ki > 25000 nM T11211 C34FBN 72544603 IC50 > 10000 nM T11211 CFN73T 72704511 IC50 = 290 nM T11211 CLA3Y9 72710581 Ki = 239 nM T11211 C7UDN2 72710911 IC50 = 30100 nM T11211 C3POU0 72736045 Ki = 243 nM T11211 C8R1CQ 72950535 EC50 = 28130 nM T11211 CJZW17 72950698 EC50 = 12680 nM T11211 CK3RU8 73347518 IC50 = 1900 nM T11211 C21BPD 73348897 IC50 = 3548.13 nM T11211 C4YJ6D 73443127 IC50 = 316.2 nM T11211 C2C8EY 76311184 Ki = 3000 nM T11211 CLDK62 76311185 Ki = 600 nM T11211 C42ZLK 76311186 Ki = 4100 nM T11211 C0J7TB 76311187 Ki = 2100 nM T11211 CDBK28 76314789 Ki = 3000 nM T11211 CV0Q6D 76314790 Ki = 3000 nM T11211 CD06UJ 76314791 Ki = 1400 nM T11211 C9X1PW 76318388 Ki = 3000 nM T11211 CLG36A 76318389 Ki = 1300 nM T11211 C6QCD8 76318390 Ki = 3600 nM T11211 CZ8M6Q 76318391 Ki = 11000 nM T11211 CWYC26 76318392 Ki = 2000 nM T11211 C3E1HS 76318393 Ki = 200 nM T11211 C49JFZ 76322066 Ki = 4000 nM T11211 CBLS90 76322067 Ki = 7000 nM T11211 C49VZL 76322068 Ki = 3000 nM T11211 CQUW30 76322069 Ki = 2100 nM T11211 CDX1Y6 76322070 Ki = 10000 nM T11211 CHLY70 76325684 Ki = 1900 nM T11211 CP9OB2 76325685 Ki = 13000 nM T11211 CKDC92 76325686 Ki = 2700 nM T11211 COQ4I8 76329255 Ki = 4100 nM T11211 CKY5X3 76329256 Ki = 12000 nM T11211 CU9EA3 76332906 Ki = 2300 nM T11211 C0K2UJ 76332907 Ki = 2500 nM T11211 CQ7BL1 76332908 Ki = 32000 nM T11211 CZ7X4N 76332909 Ki = 2200 nM T11211 CPM2F6 76332910 Ki = 56000 nM T11211 CB1W6D 76332911 Ki = 3000 nM T11211 C6GUL4 76336517 Ki = 2300 nM T11211 CMW24P 76336518 Ki = 400 nM T11211 CKFZ96 76336519 Ki = 1700 nM T11211 CAH3R2 78319202 IC50 = 49000 nM T11211 C8OSE1 78319203 IC50 = 45000 nM T11211 C35VEY 78319204 IC50 = 40000 nM T11211 C1G0FL 82371100 IC50 = 3670 nM T11211 C3RHG9 85468997 EC50 = 190 nM T11211 CK20QY 86276216 EC50 = 2.5 nM T11211 CIU65X 86280440 Ki = 232 nM T11211 CXEN05 86287624 IC50 = 15.41 nM T11211 CG28YT 86605033 IC50 = 7.5 nM T11211 CV2JZ1 86697032 Ki = 43.3 nM T11211 CT50AL 87539277 IC50 > 1000 nM T11211 CY05IC 87733533 IC50 > 1000 nM T11211 C9EH7I 89500376 Ki = 5.21 nM T11211 C0EQS7 89501406 EC50 = 4.88 nM T11211 C8JG7O 89510193 EC50 = 0.0398 nM T11211 CP91ZD 89541678 Ki = 481.8 nM T11211 CR3W1F 89541680 Ki = 257 nM T11211 CT56PQ 89542198 Ki = 95.3 nM T11211 C1N6FP 89553258 Ki = 126.1 nM T11211 CVJG67 89553307 Ki = 33.8 nM T11211 C4JM1T 89553308 Ki = 215.4 nM T11211 CK5D1A 90395281 IC50 = 13000 nM T11211 CW6E5N 90655068 EC50 = 1.8 nM T11211 CCL56B 90655069 EC50 = 1.7 nM T11211 C7KD0Q 90655070 EC50 = 0.15 nM T11211 C8SU6Z 90655071 EC50 = 0.074 nM T11211 C2E1PI 90655072 EC50 = 0.4 nM T11211 C7YCR3 90655073 EC50 = 1.1 nM T11211 CM7I3P 90655074 EC50 = 0.06 nM T11211 C0S3WI 90655075 EC50 = 0.039 nM T11211 C37STG 90655076 EC50 = 7.6 nM T11211 CTVS25 90655077 EC50 = 17.1 nM T11211 CQ7GH9 90655078 EC50 = 2.9 nM T11211 CSQ8X5 90655079 EC50 = 0.61 nM T11211 CK51SM 90655080 EC50 = 0.28 nM T11211 C0OQ6T 90655081 EC50 = 0.25 nM T11211 CC2LT8 90655082 EC50 = 0.11 nM T11211 CP3VA1 90655083 EC50 = 689 nM T11211 CDK7A2 90655084 EC50 = 37.4 nM T11211 CN5D4R 90655085 EC50 = 14.8 nM T11211 CVIO18 90655086 EC50 = 3.4 nM T11211 CY2R5Q 90655087 EC50 = 275 nM T11211 CQ1F3H 90655088 EC50 = 6.1 nM T11211 C40DRC 90655089 EC50 = 0.34 nM T11211 CO09NQ 90655090 EC50 = 1.8 nM T11211 CX57EB 90655091 EC50 = 8.6 nM T11211 CI3YE2 90655092 EC50 = 6.8 nM T11211 CYO4Q2 90655093 EC50 = 7.2 nM T11211 C6VZ7X 90656360 IC50 > 10000 nM T11211 CNCB43 90656361 IC50 > 10000 nM T11211 CYR64B 91754488 IC50 = 170 nM T11211 CY59AC 95555777 IC50 = 160 nM T11211 CD0ON3 101883236 IC50 = 3580 nM T11211 C4N0MB 101883242 IC50 = 770 nM T11211 C0GYL7 102364501 IC50 = 840 nM T11211 CJ98HE 112777808 EC50 > 25000 nM T11211 CN5ZQ2 117629963 EC50 = 1650 nM T11211 C8F0CN 117967617 EC50 = 12000 nM T11211 C9GM4N 117968554 EC50 = 11100 nM T11211 C2D8MQ 117976829 EC50 = 3100 nM T11211 CW27MY 118063735 EC50 > 30000 nM T11211 CU37BH 118233211 Ki = 14.1 nM T11211 C70XEJ 118310050 IC50 = 180 nM T11211 CS8TG5 118310052 IC50 = 3020 nM T11211 CL58OA 118310053 IC50 = 270 nM T11211 C17XUS 118310054 IC50 = 220 nM T11211 CD7EK4 118310055 IC50 = 3560 nM T11211 C8ZB0V 118310056 IC50 = 230 nM T11211 C8YL5A 118310059 IC50 = 1190 nM T11211 CR21JK 118314640 IC50 = 250 nM T11211 CS3UR5 118314642 IC50 = 2580 nM T11211 CN43EZ 118314645 IC50 = 1740 nM T11211 C50PAC 118314647 IC50 = 700 nM T11211 CQ94NF 118314654 IC50 = 440 nM T11211 CJ65NZ 118314655 IC50 = 3560 nM T11211 CCF0N9 118314665 IC50 = 960 nM T11211 CYCF19 118314668 IC50 = 570 nM T11211 CT3HC7 118314670 IC50 = 1280 nM T11211 CLS7C1 118707978 Ki > 50000 nM T11211 C9LV0M 118707979 Ki > 50000 nM T11211 CY3D4B 118708589 IC50 = 8090 nM T11211 C8UY3L 118708590 IC50 = 9440 nM T11211 CY2J0Z 118708591 IC50 = 5200 nM T11211 C6E7GC 118708592 IC50 = 5480 nM T11211 CYM7R6 118708593 IC50 = 3060 nM T11211 CU8A3E 118708594 IC50 = 5450 nM T11211 C8IXT1 118708595 IC50 = 1650 nM T11211 CJV5F9 118708596 IC50 = 1770 nM T11211 CP49YN 118708597 IC50 = 1200 nM T11211 C7IWN4 118708598 IC50 = 1100 nM T11211 C0M9JL 118708599 IC50 = 850 nM T11211 C94TNF 118708600 IC50 = 1000 nM T11211 CDQ7J4 118708601 IC50 = 500 nM T11211 CCH2A3 118708602 IC50 = 430 nM T11211 CW41DN 118710795 IC50 = 1730 nM T11211 CFNH62 118710796 IC50 = 2610 nM T11211 CC2H4E 118714881 IC50 > 10000 nM T11211 CC01IF 118717325 IC50 = 83800 nM T11211 CQU2Z0 118732596 IC50 = 39.8 nM T11211 CZO48M 118732597 IC50 = 29.3 nM T11211 CXQY05 118732598 IC50 = 233 nM T11211 C2VK0B 118732599 IC50 = 2650 nM T11211 C1DY9P 118732600 IC50 = 2040 nM T11211 C9RH8V 121350767 IC50 = 3100 nM T11211 C9Q6WA 121350771 IC50 = 710 nM T11211 CG13LX 122178361 IC50 = 3400 nM T11211 C8DM9B 122180597 Ki = 40.6 nM T11211 C0C6NJ 122180598 Ki = 797.6 nM T11211 C8X5FP 122180599 Ki = 514.5 nM T11211 C1L4JM 122180600 Ki = 235.9 nM T11211 CHC0I6 122180602 Ki = 584.6 nM T11211 C6GF7V 122180603 Ki = 575.6 nM T11211 CH8QE1 122180846 Ki = 11.9 nM T11211 CCV15M 122186565 IC50 = 2400 nM T11211 C7V6LB 122186567 IC50 = 620 nM T11211 CY18QG 122186737 Ki = 4140 nM T11211 C0OR2H 122186738 Ki = 6120 nM T11211 CU0Y8B 122186739 Ki = 4060 nM T11211 CWF0Q4 122186740 Ki = 1120 nM T11211 CBE6Q8 122186741 Ki = 231 nM T11211 CX13DR 122186742 Ki = 684 nM T11211 CJ74HX 122186743 Ki = 905 nM T11211 C05VWL 122186744 Ki = 1130 nM T11211 CNX5H4 122186745 Ki = 697 nM T11211 CQ6BG8 122186747 Ki = 91 nM T11211 CH8O2M 122186748 Ki = 401 nM T11211 C4LRN1 122186749 Ki = 496 nM T11211 CCU09A 122191896 IC50 = 530 nM T11211 C9DXI2 122191898 IC50 = 1010 nM T11211 CB95XH 122191900 IC50 = 1660 nM T11211 CAMQ21 122191901 IC50 = 3710 nM T11211 CI96FE 122191902 IC50 = 1950 nM T11211 C94EOP 122191903 IC50 = 9020 nM T11211 CH8G2I 122191904 IC50 = 1380 nM T11211 CGH1S3 122191905 IC50 = 3760 nM T11211 CH2L7K 122191906 IC50 = 180 nM T11211 CC5S2M 122191907 IC50 = 920 nM T11211 CN9C2T 122192181 IC50 > 31622.78 nM T11211 CY7PA4 122192281 Ki = 8 nM T11211 C9QV1Y 122192282 Ki = 1600 nM T11211 C6WL8N 122192283 IC50 = 22 nM T11211 C56NUY 122192284 Ki = 31 nM T11211 CVO26Q 122192285 Ki = 3 nM T11211 C72DZH 122192286 IC50 = 34 nM T11211 C8CPQ9 122192287 Ki = 31 nM T11211 CXT0C5 122192288 IC50 = 6 nM T11211 CB31UD 122192289 Ki = 12 nM T11211 C4DVB5 122192290 IC50 = 1 nM T11211 CC9T1P 122192291 Ki = 1 nM T11211 CM8BR7 122192292 Ki = 2 nM T11211 CTI2V5 122192293 Ki = 1.7 nM T11211 CMC4P7 122197406 EC50 = 2.8 nM T11211 CXZ8T3 122197407 Ki = 3.1 nM T11211 C8U0YD 122512150 EC50 = 16100 nM T11211 C9EJ3D 122512151 EC50 > 25000 nM T11211 C7EVD2 122512153 EC50 = 12700 nM T11211 C5NTP8 122512155 EC50 = 2700 nM T11211 C4ZCJ5 122512159 EC50 = 7700 nM T11211 CAF4G0 122512161 EC50 > 25000 nM T11211 CKJH03 122512162 EC50 > 25000 nM T11211 CSQL81 122512166 EC50 = 7200 nM T11211 CO8BK9 122512168 EC50 = 18400 nM T11211 CUBT32 122512169 EC50 = 11100 nM T11211 CC0YK8 122512171 EC50 > 25000 nM T11211 CDLP71 122512175 EC50 > 25000 nM T11211 CKHD34 122512178 EC50 = 10800 nM T11211 CGN3D8 122527240 EC50 > 25000 nM T11211 CAT9G6 122527241 EC50 = 14700 nM T11211 C45SLP 122527242 EC50 = 16600 nM T11211 CGJO26 122531962 EC50 > 25000 nM T11211 CAN89H 122534294 EC50 = 2900 nM T11211 CSX95E 122640053 IC50 = 99 nM T11211 C5C0WL 122640061 IC50 = 37 nM T11211 CTI21U 122640063 IC50 = 64 nM T11211 CZ3K5G 122640065 Ki = 135 nM T11211 CN4Z3Q 122640071 IC50 = 45 nM T11211 C9X8ZE 122640074 Ki = 86 nM T11211 CE3A5F 122640078 IC50 = 127 nM T11211 C3A7PB 122640079 IC50 = 157 nM T11211 C2AQM7 122640083 IC50 = 85 nM T11211 C17EFK 122640084 Ki = 71 nM T11211 C7RL0P 122640088 IC50 = 130 nM T11211 C4F8JN 122640093 IC50 = 32 nM T11211 CF09JD 122640094 IC50 = 142 nM T11211 CJ1I9O 122640101 IC50 = 94 nM T11211 C37UBT 122640109 Ki = 133 nM T11211 CQ0WH1 122640117 Ki = 316 nM T11211 COT0Z9 122640118 IC50 = 39 nM T11211 C5NC3G 122640121 IC50 = 142 nM T11211 CZ4F5V 122640122 IC50 = 101 nM T11211 CK27OF 122640126 IC50 = 59 nM T11211 CRX1K5 122640131 Ki = 84 nM T11211 C9YZ0T 122640134 Ki = 204 nM T11211 CEN27X 122640138 IC50 > 10000 nM T11211 C5MXG2 122640139 IC50 = 126 nM T11211 CIX05D 122640140 Ki = 294 nM T11211 CA58HO 122640144 Ki = 68 nM T11211 C81VHX 122640145 Ki = 124 nM T11211 CZ3EI2 122640149 IC50 = 598 nM T11211 C2EQY4 122640156 IC50 = 85 nM T11211 C7MXJ0 122640160 IC50 = 234 nM T11211 C0QJ7B 122640163 IC50 = 88 nM T11211 CLB1H3 122640167 Ki = 47 nM T11211 CVF5G3 122650648 IC50 = 48 nM T11211 C97BZD 122651003 IC50 = 686 nM T11211 C8EZ6C 122651049 IC50 = 972 nM T11211 CX6I3E 126505404 Ki = 62 nM T11211 CGWK72 127048374 EC50 = 7.943 nM T11211 CJNA49 127048375 EC50 = 10000 nM T11211 C9L5TC 127048376 EC50 = 0.1585 nM T11211 CR3H9B 127048377 EC50 = 1.585 nM T11211 CS6PF7 127048378 EC50 = 31.62 nM T11211 C0NGD5 127048379 EC50 = 39.81 nM T11211 C7MN5C 127048380 EC50 = 2511.89 nM T11211 CMKG20 127048381 EC50 = 12.59 nM T11211 CL2G9I 127048724 EC50 = 1.585 nM T11211 CTAO91 127049032 EC50 = 12.59 nM T11211 CXA3Y6 127049350 EC50 = 3.162 nM T11211 CHNV46 127049374 EC50 = 15.85 nM T11211 C0SX8P 127049375 EC50 = 3.981 nM T11211 C1Y3IL 127049376 EC50 = 1.585 nM T11211 CD9LF5 127049693 EC50 = 19.95 nM T11211 CI6C2H 127049715 EC50 = 0.2512 nM T11211 C1ZEF2 127049716 EC50 = 0.03162 nM T11211 CKL54Q 127049717 EC50 = 0.1995 nM T11211 CJ0IL6 127049718 EC50 = 15.85 nM T11211 CMYW48 127050010 EC50 = 1.995 nM T11211 CO4PX6 127050295 EC50 = 3.981 nM T11211 CKNE38 127050356 EC50 = 5.888 nM T11211 CA9N5D 127050357 EC50 = 0.5012 nM T11211 CN26ZR 127050358 EC50 = 0.2512 nM T11211 C6RJ1U 127050609 EC50 = 63.1 nM T11211 CGH85U 127050670 EC50 = 5.623 nM T11211 CQ6M5O 127050671 EC50 = 2.884 nM T11211 CVK37R 127050944 EC50 = 0.3981 nM T11211 C45PWI 127050978 EC50 = 15.85 nM T11211 C8WTG6 127050979 EC50 = 1.259 nM T11211 C3OQ4S 127050980 EC50 = 1.259 nM T11211 C02GPQ 127050981 EC50 = 1.995 nM T11211 CA49NU 127050982 EC50 = 2.512 nM T11211 CI29LO 127050983 EC50 = 10.47 nM T11211 C4V8AP 127051245 EC50 = 0.631 nM T11211 CNS96C 127051246 EC50 = 3.162 nM T11211 CG75RD 127051247 EC50 = 19.95 nM T11211 CRPH62 127051248 EC50 = 0.7943 nM T11211 CKH8M3 127051249 EC50 = 0.1995 nM T11211 CU8BJ5 127051250 EC50 = 79.43 nM T11211 CA2ZR6 127051251 EC50 = 3.981 nM T11211 CL48ZN 127051252 EC50 = 79.43 nM T11211 C8BVP3 127052745 EC50 = 1.995 nM T11211 CFH3G1 127053068 EC50 = 19.95 nM T11211 CQ7M9C 127053069 EC50 = 3.981 nM T11211 C89WDR 127053070 EC50 = 158.49 nM T11211 C86RXZ 127053071 EC50 = 1.585 nM T11211 CA79BG 127053072 EC50 = 3.162 nM T11211 CJM83P 127053073 EC50 = 2.512 nM T11211 CDN2P8 127053074 EC50 = 0.7943 nM T11211 COR0W5 127053075 EC50 = 0.1995 nM T11211 CY0WZ9 129295280 EC50 = 224 nM T11211 C65RIZ 129295282 EC50 > 2500 nM T11211 CM62UE 129295287 EC50 > 2500 nM T11211 CR23ZG 129295311 IC50 = 642 nM T11211 C2LVO7 129295370 IC50 = 3146 nM T11211 CTI04S 129295372 IC50 = 1295 nM T11211 C4G2ID 129304679 EC50 > 2500 nM T11211 CGK48C 129304682 EC50 > 2500 nM T11211 CEVZ49 129304683 EC50 > 2500 nM T11211 CM4LD6 129304687 EC50 > 2500 nM T11211 C6XAZ5 129304688 EC50 > 2500 nM T11211 C85QXL 129304691 EC50 > 2500 nM T11211 CR3YV9 129304702 EC50 > 2500 nM T11211 CS2UB8 129304733 EC50 > 2500 nM T11211 COU93J 129304741 EC50 > 2500 nM T11211 C7K2IE 129304748 EC50 > 2500 nM T11211 C2GJ8T 129304757 EC50 > 2500 nM T11211 C7MRB5 129304758 IC50 = 129 nM T11211 CN0UA7 129304771 EC50 > 2500 nM T11211 CBSJ31 129304830 EC50 > 2500 nM T11211 C1H0UX 129304861 EC50 > 2500 nM T11211 C7ZI4T 131337559 EC50 = 573.2 nM T11211 CS3C8P 132471744 EC50 = 0.34 nM T11211 CN9DL4 134132030 IC50 = 68 nM T11211 CG9WU7 134132399 Ki = 48 nM T11211 CU58EQ 134135199 Ki = 5 nM T11211 CX93QK 134135812 IC50 = 110 nM T11211 C53UTO 134137062 IC50 = 43 nM T11211 C9TG2N 134137487 IC50 > 1000 nM T11211 CSX58U 134139437 IC50 < 30 nM T11211 C75NRQ 134141877 IC50 < 30 nM T11211 C62SVR 134142119 IC50 = 250 nM T11211 CLI48U 134143743 IC50 = 330 nM T11211 CWRJ15 134147087 IC50 = 230 nM T11211 C8K0XJ 134147090 IC50 < 30 nM T11211 CJE92T 134149144 Ki = 8 nM T11211 CQ61SB 134150479 IC50 = 78 nM T11211 CDX75O 134152551 IC50 < 30 nM T11211 C2JV5X 134153768 IC50 = 350 nM T11211 C4FLQ5 134157355 IC50 = 560 nM T11211 C1UP3S 134157845 IC50 < 30 nM T11211 C30HIQ 134415607 IC50 = 359 nM T11211 C3Y2NT 134415609 IC50 = 354 nM T11211 CQ53DW 134415610 EC50 > 2500 nM T11211 CO32XF 134415624 IC50 = 208 nM T11211 CRP1C4 134415742 IC50 = 175 nM T11211 C1U9HD 134415745 IC50 = 263 nM T11211 CB09XQ 134415864 EC50 = 1142 nM T11211 CU6Y5D 134415868 IC50 = 1005 nM T11211 C1GY2T 135156251 EC50 > 10000 nM T11211 CTL4P3 135403572 IC50 = 50000 nM T11211 CY8U6E 135459005 IC50 = 12400 nM T11211 CJA70N 135459106 IC50 = 11100 nM T11211 C34JMK 135571931 IC50 = 33200 nM T11211 C5MXO2 136000568 Ki = 430 nM T11211 CM6OX5 136000656 Ki = 290 nM T11211 CZ2D6U 136059148 Ki = 1000 nM T11211 C6HOU3 136059149 Ki = 90 nM T11211 CE1G9O 136059150 Ki = 2800 nM T11211 C7LSN6 136088946 Ki = 1500 nM T11211 CX63JK 137631530 IC50 = 6.8 nM T11211 C9H1WV 137632762 EC50 = 1517.7 nM T11211 COW6F1 137633683 EC50 = 980 nM T11211 C1PMS4 137634112 IC50 = 2.9 nM T11211 COI80Z 137634236 IC50 > 1000 nM T11211 C5EDV3 137635222 IC50 = 25820 nM T11211 CW4V8D 137635242 EC50 = 17.8 nM T11211 CB4TC2 137636774 IC50 = 8170 nM T11211 C8KW3H 137637301 IC50 = 47.6 nM T11211 CBFS94 137637469 EC50 = 1136.4 nM T11211 C1KCY9 137639290 IC50 = 4.9 nM T11211 CPD87Y 137639726 IC50 > 1000 nM T11211 CK6RM4 137640380 IC50 = 21510 nM T11211 CVW6U9 137640542 EC50 = 15.2 nM T11211 CGJ4R8 137640796 IC50 = 166.9 nM T11211 CYG4M9 137641824 EC50 = 1.7 nM T11211 C91MCO 137643639 EC50 = 1450.3 nM T11211 CL0F4T 137644265 IC50 = 22590 nM T11211 CMH4Q7 137644499 IC50 = 18750 nM T11211 C4RUL8 137644639 IC50 = 5960 nM T11211 C3LE1F 137644659 EC50 = 1341.7 nM T11211 C28JCE 137646631 IC50 = 6032 nM T11211 C49OST 137647704 IC50 = 14 nM T11211 CFGR61 137648154 IC50 = 27960 nM T11211 C30ZJF 137648477 IC50 = 316.23 nM T11211 C24RKO 137648986 EC50 = 0.17 nM T11211 CF9QP1 137649447 IC50 = 1465.9 nM T11211 C2FPL5 137651323 IC50 = 3.7 nM T11211 C7VOQ6 137652389 IC50 = 13170 nM T11211 CI75TS 137653348 EC50 = 0.14 nM T11211 CO92KL 137654415 IC50 = 794.33 nM T11211 CM7X0Z 137654630 EC50 = 229.1 nM T11211 CP8K6X 137655620 IC50 = 5.5 nM T11211 CZX69U 137656474 EC50 = 5.3 nM T11211 CV9GO0 137657324 EC50 = 391 nM T11211 C3O7HB 137658245 IC50 = 10960 nM T11211 CEL81T 137658776 EC50 > 10000 nM T11211 CPV2Q5 137659321 EC50 = 233 nM T11211 CHW01P 137662044 IC50 = 7780 nM T11211 C7EKA2 138911324 IC50 = 912 nM T11211 C96ONI 141538600 IC50 = 561 nM T11211 CR6Y2I 141538601 IC50 = 1452 nM T11211 CR5Y9P 145949269 EC50 = 13 nM T11211 CW3Y0H 145949340 IC50 > 20000 nM T11211 CP5U7Q 145949975 EC50 > 2500 nM T11211 COKU96 145950643 EC50 = 1.5 nM T11211 CPK5U1 145951022 IC50 = 300 nM T11211 CJX58K 145951453 IC50 = 83800 nM T11211 CKT24R 145951943 IC50 = 1800 nM T11211 CD49VI 145953389 EC50 > 2500 nM T11211 CL05IG 145956989 IC50 = 7390 nM T11211 CU19EN 145958055 EC50 = 54 nM T11211 C5U3JV 145958117 EC50 = 30 nM T11211 CORP09 145958365 EC50 > 2500 nM T11211 CR6T8S 145959457 EC50 > 2500 nM T11211 CPQ03X 145968294 IC50 = 54 nM T11211 C1CH7Y 145968379 IC50 = 1100 nM T11211 CG57QD 145968598 IC50 = 53 nM T11211 CCE13D 145969025 IC50 = 190 nM T11211 C8YHF2 145969445 IC50 = 27 nM T11211 C7K9AC 145970643 IC50 = 190 nM T11211 CXVW37 145970907 IC50 > 10000 nM T11211 C96SNM 145978980 IC50 < 1000 nM T11211 CAI3Z5 145980066 IC50 = 1680 nM T11211 C8U7BE 145980222 IC50 = 3570 nM T11211 CKIX59 145987210 IC50 = 1420 nM T11211 CH3K6N 145989528 IC50 = 1770 nM T11211 CL0UA8 145989688 IC50 > 10000 nM T11211 CH0DY7 145989890 IC50 = 4260 nM T11211 CW70GB 145990651 IC50 = 1720 nM T11211 CC7BO9 145990706 IC50 = 5270 nM T11211 C3PU6X 145991012 IC50 = 3960 nM T11211 C7BM6C 145993790 IC50 = 2870 nM T11211 CCZ9N7 145993833 IC50 = 1640 nM T11211 CG3XW1 155187679 IC50 = 641.3 nM T11211 C30SYM 155459658 EC50 > 2500 nM T11211 CGB78J 155459666 IC50 = 2955 nM T11211 CT9B6U 155519221 IC50 = 9 nM T11211 CXE0W4 155529903 IC50 = 315 nM T11211 C9AV0G 155546681 EC50 > 100 nM T11211 C1XGF5 155546726 EC50 = 1885 nM T11211 C64VLC 155549606 EC50 = 470 nM T11211 CI3SZ0 155554274 Ki = 11 nM T11211 C8JI3Y 155562428 IC50 = 392 nM T11211 D00BLY 44157042 IC50 = 10 nM T11211 D00CDF 9824562 Ki = 4 nM T11211 D00RIX 5280443 IC50 = 5200 nM T11211 D01ETZ 261000 EC50 = 0.013 nM T11211 D01THF 44564580 IC50 = 39 nM T11211 D02CXU 44565151 IC50 = 353 nM T11211 D02RQP 6623 IC50 = 5900 nM T11211 D02UID 16734800 IC50 = 2300 nM T11211 D02ZEE 25093227 IC50 = 20.1 nM T11211 D03MQA 44564583 IC50 = 55 nM T11211 D03VQC 44564585 IC50 = 1730 nM T11211 D03WHD 16090308 IC50 = 26 nM T11211 D04KPW 44565104 IC50 = 57 nM T11211 D04PLB 11507014 IC50 = 30 nM T11211 D04QAT 43138559 IC50 = 4000 nM T11211 D04USO 11587567 IC50 = 198 nM T11211 D05FPU 44564582 IC50 = 66 nM T11211 D06BLF 18728 IC50 = 42.7 nM T11211 D06JPP 9839132 EC50 = 3 nM T11211 D06PRV 44565102 IC50 = 43 nM T11211 D06WNK 44157041 IC50 = 30 nM T11211 D06YKU 68112 IC50 = 831.76 nM T11211 D06ZZM 11673174 IC50 = 46 nM T11211 D07AHG 15521397 IC50 > 10000 nM T11211 D07GCR 44565205 IC50 = 1340 nM T11211 D07KWO 9823099 IC50 = 6500 nM T11211 D07QFN 44565152 IC50 = 5210 nM T11211 D07TVI 25093231 IC50 = 37 nM T11211 D08DHC 11608821 IC50 = 92 nM T11211 D08FZN 9903530 IC50 = 27.5 nM T11211 D08FZR 44565206 IC50 = 20 nM T11211 D08KQM 24816375 Ki = 910 nM T11211 D08QWR 616651 IC50 = 5370 nM T11211 D08RCS 44564581 IC50 = 40 nM T11211 D09OKK 9951771 Ki = 844 nM T11211 D09SJY 11715659 IC50 = 24 nM T11211 D0B2JG 43320723 IC50 = 770 nM T11211 D0B5GC 11349 IC50 = 23500 nM T11211 D0BU5X 44564584 IC50 = 441 nM T11211 D0F1SS 44605900 IC50 > 10000 nM T11211 D0FI1I 11557752 IC50 = 115 nM T11211 D0G0XB 44434099 IC50 > 1 nM T11211 D0G3IT 132581 IC50 = 15 nM T11211 D0G3TK 5280863 IC50 = 9700 nM T11211 D0G5OV 11543746 IC50 = 196 nM T11211 D0GR5L 9906282 Ki = 1230 nM T11211 D0I5YU 43138589 IC50 = 11 nM T11211 D0J7XZ 9819614 Ki = 650 nM T11211 D0L5IC 9820558 Ki = 130 nM T11211 D0L7OC 43615786 IC50 = 49 nM T11211 D0M0RS 11560224 EC50 = 0.2 nM T11211 D0O0ZC 2734580 IC50 = 3300 nM T11211 D0P0ZQ 44157043 IC50 = 89 nM T11211 D0RI6O 44397072 IC50 = 63 nM T11211 D0S0RK 10680 IC50 = 5900 nM T11211 D0S9YX 5280373 IC50 = 1600000 nM T11211 D0SP7S 5995 Ki = 0.25 nM T11211 D0T7LR 44565150 IC50 = 200 nM T11211 D0U9IR 44565202 IC50 = 123 nM T11211 D0V3UU 11178122 IC50 = 200 nM T11211 D0V5HF 94525 IC50 = 8700 nM T11211 D0VE6A 44564659 IC50 = 519 nM T11211 D0W5IF 11632731 IC50 = 410 nM T11211 D0XS0R 44433505 Ki = 8892 nM T57174 D0E3TC 44259 IC50 = 850 nM T57174 D0R2TM 5287736 IC50 = 47 nM T57174 CQR05P 11494718 IC50 = 1.8 nM T57174 CHT93E 11502159 IC50 = 4.3 nM T57174 CV63UL 67240318 IC50 > 10000 nM T57174 CG2JO7 137638433 IC50 = 0.65 nM T57174 CX5BK1 137647477 IC50 = 3.3 nM T57174 C8R0JP 137654554 IC50 = 21 nM T57174 C2MD1Q 155513187 IC50 > 10000 nM T57174 D0U8UK 11677079 IC50 = 5.4 nM T30938 D0G3DL 135398735 IC50 < 10 nM T30938 C34TOA 6436726 IC50 < 10 nM T30938 CI0RK5 57390968 IC50 = 503 nM T30938 CUL04F 57390970 IC50 = 15400 nM T30938 CSI87U 57398041 IC50 = 4400 nM T30938 C7X8OH 57401461 IC50 = 21 nM T30938 C84UFN 57403202 IC50 = 15 nM T30938 CHN6S4 136098617 IC50 = 13 nM T30938 C3PN5F 136098618 IC50 = 142 nM T30938 CFI40H 136098619 IC50 = 139 nM T86582 D00ENY 33032 IC50 = 11000 nM T86582 C9CQV1 131738 IC50 = 270000 nM T86582 C7BKY8 164701 IC50 = 100000 nM T86582 C45TML 1755783 IC50 > 300000 nM T86582 CDK9W5 1796705 IC50 > 300000 nM T86582 C8L6JU 2177697 IC50 = 22908.68 nM T86582 CRQW20 2266743 IC50 > 300000 nM T86582 CO0I2U 2266913 IC50 > 300000 nM T86582 C9HE6N 2271641 IC50 > 300000 nM T86582 CH4RP6 2271698 IC50 > 300000 nM T86582 C3SL4Y 2271738 IC50 > 300000 nM T86582 C7K9MX 2283576 IC50 = 12000 nM T86582 CB6EZ4 2285406 IC50 > 300000 nM T86582 CBW36C 2287441 IC50 > 316227.77 nM T86582 C13DLB 2289587 IC50 > 316227.77 nM T86582 CZQ83G 2289624 IC50 > 300000 nM T86582 CFG35Z 2737891 IC50 = 2290.87 nM T86582 CYR4X2 2838960 IC50 = 3630.78 nM T86582 CP4L3M 2839392 IC50 = 4000 nM T86582 CF2LE3 4133412 IC50 = 3162.28 nM T86582 CJW9P4 5506801 IC50 > 300000 nM T86582 C5PWJ3 6505351 IC50 > 300000 nM T86582 CTBZ42 6505352 IC50 = 100000 nM T86582 C64QSY 7016554 Ki = 11481.54 nM T86582 CTMP80 9920506 Ki = 22908.68 nM T86582 C2EA8S 10219727 IC50 > 1000000 nM T86582 C53YBE 10419887 Ki > 400000 nM T86582 C2PE4O 10464763 IC50 = 100000 nM T86582 C46KUE 10680281 Ki = 117489.76 nM T86582 C2WQB7 10877814 IC50 > 1000000 nM T86582 C83OPZ 10954230 IC50 > 1000000 nM T86582 C7Z6AX 10986716 IC50 > 1000000 nM T86582 C78YAI 10997729 IC50 > 1000000 nM T86582 CE80SU 11041159 IC50 > 1000000 nM T86582 CMSD95 11062853 IC50 > 1000000 nM T86582 C2TWR9 11063103 IC50 > 1000000 nM T86582 C0HT8M 11528550 Ki = 40738.03 nM T86582 CQ5H1B 11543205 Ki = 127000 nM T86582 C2QJU5 11616374 IC50 = 2000 nM T86582 CZ9V5S 11629898 Ki = 28840.32 nM T86582 C5E8BT 11651356 Ki = 47863.01 nM T86582 CV76LO 11667702 IC50 = 3800 nM T86582 C7SHB1 11745400 Ki = 10232.93 nM T86582 C0BM2Z 12047098 IC50 = 69000 nM T86582 C68AOJ 12047099 IC50 = 15000 nM T86582 C09XIT 12047100 IC50 = 16000 nM T86582 C1X3YB 16727662 IC50 > 300000 nM T86582 C6XLF5 24905646 IC50 = 3000000 nM T86582 CFI54P 24905647 IC50 > 1000000 nM T86582 CQK96U 24905648 IC50 > 3000000 nM T86582 C36NMZ 24905649 IC50 = 1000000 nM T86582 CB3T7C 24905650 IC50 = 1000000 nM T86582 C14RNW 24905651 IC50 = 3000000 nM T86582 CM1S2B 24905652 Ki = 450000 nM T86582 CUS45D 24905703 IC50 > 3000000 nM T86582 C86BUK 24905705 Ki > 3000000 nM T86582 CJ25EZ 44404580 IC50 = 300 nM T86582 C0LJ8T 44404590 IC50 = 3000 nM T86582 CJD1V7 44404611 IC50 = 700 nM T86582 CJ6ER9 44404615 IC50 = 2000 nM T86582 C4CZN1 44405320 Ki = 28840.32 nM T86582 C8TMX2 44417425 Ki = 200000 nM T86582 CYQ2S5 49782834 IC50 > 1000000 nM T86582 C94ZJF 49782835 IC50 > 100000 nM T86582 CZ5YU8 49783035 IC50 > 100000 nM T86582 CR2IM7 49910175 IC50 > 316227.77 nM T86582 CY91US 52941382 IC50 = 3.548 nM T86582 CI76TC 70688590 IC50 > 300000 nM T86582 C2J4MG 70690647 IC50 > 300000 nM T86582 C4HI0U 70789291 IC50 > 3000000 nM T86582 CP48NY 71449125 IC50 = 20000 nM T86582 C7NYC0 71449126 IC50 = 2000 nM T86582 CD03AH 71449127 IC50 = 700 nM T86582 CVST26 71450915 IC50 = 150 nM T86582 C31HCW 71450916 IC50 = 1000 nM T86582 CC15SM 71450917 IC50 = 100000 nM T86582 CBZ9D6 71450918 IC50 = 22000 nM T86582 CSO9P3 71452727 IC50 = 200 nM T86582 C23DMA 71452728 IC50 = 130 nM T86582 CE0A3V 71452729 IC50 = 6000 nM T86582 CRKN62 71452730 IC50 = 2900 nM T86582 C8X4VU 71454504 IC50 = 200 nM T86582 COUY80 71454505 IC50 = 100 nM T86582 C8QW6K 71454506 IC50 = 1000 nM T86582 CKWF24 71454507 IC50 = 6000 nM T86582 CDY5K2 71456248 IC50 = 400 nM T86582 C9O7LC 71456249 IC50 = 100 nM T86582 C1HJF2 71458054 IC50 = 300 nM T86582 C3P0MQ 71461655 IC50 = 3000 nM T86582 C0P4NT 71574743 IC50 > 300000 nM T86582 CGH79X 71574744 IC50 > 300000 nM T86582 COC8W2 71574746 IC50 > 300000 nM T86582 C5U9HZ 71574747 IC50 > 300000 nM T86582 C35BOJ 71574834 IC50 > 1000000 nM T86582 CNVG02 71574836 IC50 = 100000 nM T86582 C2JS0I 71574837 IC50 = 200000 nM T86582 CV5IT8 71574838 IC50 > 1000000 nM T86582 CL9BJ8 71574839 IC50 > 1000000 nM T86582 CCS4T2 71574840 IC50 > 1000000 nM T86582 CM5Z0I 71574841 IC50 > 300000 nM T86582 C3Z0TH 73348758 Ki = 200000 nM T86582 C8DGU5 90480101 IC50 > 1000000 nM T86582 CEH82V 90480134 IC50 > 1000000 nM T86582 CT2KF1 127030385 IC50 > 300000 nM T86582 CX95LC 127030386 IC50 > 300000 nM T86582 C8TS1X 127030387 IC50 > 300000 nM T86582 CF6NI8 127031290 IC50 > 300000 nM T86582 C2V5PM 132820245 IC50 = 31 nM T86582 CC54HS 134131748 IC50 = 31622.78 nM T86582 CM8O9I 134131963 IC50 = 794.33 nM T86582 C26CTG 134132565 IC50 = 199526.23 nM T86582 CGXV98 134133631 IC50 = 9332.54 nM T86582 C1ZAB4 134134123 IC50 = 70000 nM T86582 CZ2WH5 134134813 IC50 = 4000 nM T86582 CT3MU6 134135313 IC50 = 300000 nM T86582 CTL6A4 134135682 IC50 = 49000 nM T86582 C0MJT1 134136786 IC50 = 100000 nM T86582 CA40DU 134137403 IC50 = 12882.5 nM T86582 C1L9UX 134139672 IC50 = 1700 nM T86582 CC24GI 134139698 IC50 > 1000000 nM T86582 CTSA19 134139982 IC50 = 2500 nM T86582 CWS62H 134140412 IC50 = 43651.58 nM T86582 C5QIB1 134140490 IC50 = 63000 nM T86582 CT4QN8 134141720 IC50 = 8800 nM T86582 CJF5X7 134143016 IC50 = 300000 nM T86582 C4CT5L 134144465 IC50 = 1949.84 nM T86582 CL0EA9 134144947 IC50 = 16000 nM T86582 COM76W 134147363 IC50 > 300000 nM T86582 C9Q2JY 134147568 IC50 = 2300 nM T86582 CS38BI 134147884 IC50 = 3800 nM T86582 CP10YS 134148109 IC50 = 100000 nM T86582 CTPS85 134149212 IC50 = 2700 nM T86582 COP15G 134149427 IC50 = 2238.72 nM T86582 C6HQS8 134149488 IC50 = 794.33 nM T86582 CTH41F 134149576 IC50 = 18000 nM T86582 CQ8R9N 134149841 IC50 = 64565.42 nM T86582 C10RSO 134150446 IC50 > 300000 nM T86582 C9N0CQ 134152035 IC50 = 300000 nM T86582 C5SN8C 134152143 IC50 = 350 nM T86582 C3RAO8 134153858 IC50 = 380 nM T86582 CI3HS7 134155673 IC50 = 316.23 nM T86582 CVT7Q4 134157558 IC50 = 1600 nM T86582 CHK48B 137643975 IC50 > 1000000 nM T86582 C6J8RH 137658224 IC50 > 1000000 nM T86582 CS1X0H 145952067 IC50 = 6.1 nM T86582 C2X6ST 145952092 IC50 = 1659.59 nM T86582 CRXG02 145952717 IC50 = 2691.53 nM T86582 CZD62V 145953140 IC50 = 3000 nM T86582 C5SH4V 145953224 IC50 = 99000 nM T86582 C63MDC 145954707 IC50 = 20.89 nM T86582 C87HDC 145955435 IC50 = 6900 nM T86582 CT3H6G 145955563 IC50 = 1600 nM T86582 CIN7D3 145955863 IC50 = 1380.38 nM T86582 CZ7N3B 145956590 IC50 = 620 nM T86582 CFZK42 145957754 IC50 = 1200 nM T86582 CEX81Q 145958688 IC50 = 87000 nM T86582 C6BP3Z 145959256 IC50 = 2200 nM T86582 C8DIJ6 145960111 IC50 = 3400 nM T86582 CET93L 145971223 IC50 = 1.259 nM T86582 CGF5S1 145971489 IC50 = 29000 nM T86582 C30JVP 145971753 IC50 = 1258.93 nM T86582 CI04HT 145972021 IC50 = 11.75 nM T86582 C18GNB 145973375 IC50 = 10.72 nM T86582 CK7UW9 155519942 IC50 > 300000 nM T86582 C0Y9UF 155520160 IC50 > 300000 nM T86582 C52DFC 155524441 IC50 = 10715.19 nM T86582 C4IWE9 155525454 IC50 > 316227.77 nM T86582 CHJ5G1 155527881 IC50 > 316227.77 nM T86582 C9Z2ME 155529757 IC50 = 38000 nM T86582 CN1S4G 155530850 IC50 > 316227.77 nM T86582 C7HOI6 155533200 IC50 > 300000 nM T86582 CG65QS 155536541 IC50 = 34673.69 nM T86582 CX3ED4 155538143 IC50 > 300000 nM T86582 C4J3DC 155541203 IC50 = 100000 nM T86582 CD4B0V 155542542 IC50 > 300000 nM T86582 C87POT 155548017 IC50 > 300000 nM T86582 CPQM13 155555116 IC50 > 300000 nM T86582 CV9R4S 155557780 IC50 > 316227.77 nM T86582 C6NAQ5 155561202 IC50 > 300000 nM T86582 CF9YI6 155564787 IC50 > 300000 nM T86582 CFN45I 155565203 IC50 > 300000 nM T86582 CCK6T7 155565355 IC50 = 15848.93 nM T86582 D02JJX 11531745 IC50 = 5000 nM T86582 D03RGP 1221 IC50 > 1000000 nM T86582 D03UIR 24905704 IC50 = 1000000 nM T86582 D04XZP 107883 IC50 > 3000000 nM T86582 D07GUB 5311218 IC50 = 1621.81 nM T86582 D09HET 11622683 IC50 = 51000 nM T86582 D0F5SO 11369932 IC50 = 300 nM T86582 D0JT2N 443239 IC50 = 3890.45 nM T86582 D0OT9B 5960 IC50 = 9300 nM T86582 D0X3CF 442879 IC50 > 500000 nM T71398 D06FJO 12555 EC50 = 1020 nM T71398 CKLS40 3976 IC50 = 1000 nM T71398 CUTF63 3777682 IC50 = 37000 nM T71398 CU8IN9 11500273 IC50 > 1000000 nM T71398 C9NKV0 11580959 IC50 > 500000 nM T71398 CFPQ26 11594699 IC50 > 500000 nM T71398 C3CL4Y 11595348 IC50 > 500000 nM T71398 C4H5TI 11609518 IC50 > 500000 nM T71398 CFX34A 11624321 IC50 > 1000000 nM T71398 CJF72V 44407649 EC50 = 21900 nM T71398 C81BOG 66633232 EC50 = 290 nM T71398 CK09FD 68084651 EC50 = 1500 nM T71398 CQN01H 68111977 EC50 = 900 nM T71398 C9ND3S 68111995 EC50 = 160 nM T71398 CNJ02Q 68642181 EC50 = 500 nM T71398 CHVZ27 68642285 EC50 = 590 nM T71398 CN1YW0 68642339 EC50 = 240 nM T71398 CC3U8O 68642353 EC50 = 350 nM T71398 C6KP5T 68643387 EC50 = 190 nM T71398 C0P5GC 71604425 EC50 = 370 nM T71398 CIJ48C 71620788 EC50 = 530 nM T71398 CI0K1A 71620794 EC50 = 380 nM T71398 CV84XJ 71621106 EC50 = 240 nM T71398 C6EPF3 71622159 EC50 = 730 nM T71398 C5H8KV 71622289 EC50 = 320 nM T71398 C9HCR4 71622563 EC50 = 880 nM T71398 C6ZO9E 73388392 EC50 = 280 nM T71398 C9U2YG 118962888 EC50 = 1500 nM T71398 CDWR07 118971275 EC50 = 180 nM T67363 D0BN9X 60947 IC50 = 62000 nM T67363 D0C4RB 36314 IC50 = 34 nM T67363 D01TJY 53340771 IC50 = 3.7 nM T67363 D09ZXO 176873 IC50 = 0.54 nM T67363 D02VIP 9955461 Ki = 0.9 nM T67363 D04TKP 9913429 IC50 = 0.7 nM T67363 D08CQL 164393 Ki = 3.5 nM T67363 D08LIG 153986 IC50 > 3 nM T67363 D0B9SR 9868426 IC50 = 0.15 nM T67363 D0K0NP 9812185 IC50 > 10000 nM T67363 D0LT1S 9823503 Ki = 2 nM T67363 D0N0BI 5491394 IC50 > 50000 nM T67363 D0P8JX 177831 IC50 > 5 nM T67363 D0S3RB 216230 IC50 > 50000 nM T67363 C9F3EI 19933 IC50 = 148600 nM T67363 C2MO8K 29669 IC50 > 200000 nM T67363 CE19HD 132605 IC50 = 14000 nM T67363 C2VPW8 151947 IC50 = 38500 nM T67363 CDOC86 303776 IC50 = 3.4 nM T67363 CY0E5C 413785 IC50 = 66900 nM T67363 CX1M9K 425841 IC50 = 127200 nM T67363 CC86KB 492972 IC50 = 1.1 nM T67363 C8WOG6 1010333 IC50 = 137000 nM T67363 CS69ZF 1071025 EC50 = 1.3 nM T67363 CR1G2H 1231102 IC50 = 240 nM T67363 C5KJD8 1255325 IC50 = 132000 nM T67363 CS3V8A 1809763 IC50 = 24 nM T67363 CMT4H7 1845776 IC50 = 30 nM T67363 COX94S 2729955 IC50 = 97300 nM T67363 CFR0N1 2730204 IC50 > 200000 nM T67363 CZ06VQ 2730227 IC50 = 87300 nM T67363 CBVQ87 2730238 IC50 = 100200 nM T67363 CKM64H 2730548 IC50 = 39500 nM T67363 CSAN34 2943054 IC50 > 200000 nM T67363 CXTG90 2969603 IC50 > 200000 nM T67363 C2E9ZX 3080994 IC50 = 4100 nM T67363 C1TH9D 3126575 IC50 = 53500 nM T67363 CU1XL0 3551223 IC50 = 162100 nM T67363 CE05TF 3924471 IC50 = 180400 nM T67363 C3YM0T 4190840 IC50 = 101400 nM T67363 C9STE1 4559036 IC50 = 605 nM T67363 C5T2IQ 4609178 IC50 = 178100 nM T67363 C4H7BF 5280759 IC50 = 5.97 ug.mL-1 T67363 CHE1J8 6148173 IC50 = 18 nM T67363 C8GZR2 6342932 IC50 > 200000 nM T67363 CC2J1B 6342934 IC50 > 200000 nM T67363 CY7WS4 9799158 IC50 = 40 nM T67363 CU7VY5 9800226 IC50 = 0.8 nM T67363 CS40VO 9802158 IC50 = 0.1 nM T67363 C86OSU 9802663 IC50 = 175 nM T67363 CH19JX 9804758 IC50 = 8 nM T67363 C2SLI5 9805222 IC50 = 2 nM T67363 CJHC15 9807081 Ki = 1 nM T67363 C26JYN 9807321 Ki = 90 nM T67363 C68UYS 9808123 IC50 = 0.4 nM T67363 CVTP38 9808486 IC50 = 7 nM T67363 C8LNB0 9809477 IC50 = 2.4 nM T67363 C19PBH 9821600 IC50 > 50000 nM T67363 CO2Z6V 9822136 Ki = 3.5 nM T67363 C4LTP2 9825687 IC50 = 0.21 nM T67363 CLR39O 9826223 IC50 > 1000 nM T67363 CB0JO4 9826672 IC50 = 0.38 nM T67363 CFZP14 9826756 IC50 = 5330 nM T67363 CIF52E 9827350 IC50 = 0.04 nM T67363 C6DLN9 9827351 IC50 = 2.1 nM T67363 CQ25XG 9827352 IC50 = 0.04 nM T67363 CO16RP 9828120 IC50 = 1 nM T67363 CL6EU1 9828131 IC50 > 200000 nM T67363 CB8GP1 9828375 IC50 = 0.00092 nM T67363 C4NIC9 9828635 IC50 = 0.4 nM T67363 CJ9HV0 9828819 IC50 = 3.4 nM T67363 C1OP9I 9828979 IC50 = 16 nM T67363 C87ADQ 9830626 IC50 = 3.2 nM T67363 C31UCL 9844289 Ki = 24 nM T67363 C2UN5L 9844290 Ki = 6.5 nM T67363 CSJ1Z5 9846189 IC50 = 0.25 nM T67363 C6HAI8 9846547 IC50 = 0.22 nM T67363 CZ0AS2 9846634 IC50 = 0.7 nM T67363 CY63LZ 9846660 IC50 = 31 nM T67363 CG0H4P 9847624 IC50 = 10 nM T67363 C13KPA 9848051 Ki < 10000 nM T67363 CAR4I2 9849008 IC50 = 69 nM T67363 C13OZW 9850433 IC50 = 16 nM T67363 CB2TS1 9850990 IC50 = 1 nM T67363 CJ7SP4 9851336 IC50 = 3 nM T67363 CTM7V0 9851337 IC50 = 1.6 nM T67363 CR38MP 9853559 IC50 = 0.08 nM T67363 CEAF74 9858710 IC50 = 160 nM T67363 CVXG48 9862253 IC50 = 21 nM T67363 C6E3OL 9863046 IC50 > 100000 nM T67363 CH6NW9 9863267 IC50 = 150 nM T67363 C0G1XS 9865309 IC50 = 0.53 nM T67363 CP4U2K 9869048 IC50 = 120 nM T67363 C30BKT 9869138 IC50 = 0.3 nM T67363 CPKL80 9869692 IC50 = 20900 nM T67363 C2ZAK6 9870468 IC50 > 800000 nM T67363 CHC56Q 9870640 IC50 = 0.033 nM T67363 C9KN3Q 9872164 IC50 = 48 nM T67363 C3JA4P 9884008 IC50 > 100000 nM T67363 C5EJN9 9884317 IC50 = 470 nM T67363 CV4T6H 9885053 IC50 = 300 nM T67363 C13WGE 9886306 IC50 = 15 nM T67363 CJPG80 9891835 IC50 = 0.11 nM T67363 C49EQN 9893755 IC50 = 2 nM T67363 C6PNG8 9894403 IC50 = 3 nM T67363 C2W7NP 9894622 IC50 = 22 nM T67363 CVL6D4 9894840 IC50 = 0.9 nM T67363 CME97S 9894966 IC50 = 0.62 nM T67363 C04INH 9895205 IC50 = 230 nM T67363 CR2M8C 9901104 IC50 = 500 nM T67363 C1OY5T 9905414 IC50 = 19 nM T67363 CNX29T 9907082 IC50 = 10 nM T67363 CC6PJ4 9908437 IC50 = 29 nM T67363 C43TPN 9910543 IC50 = 32 nM T67363 C25HTY 9910653 IC50 = 33 nM T67363 CX0RQ4 9910884 Ki = 3 nM T67363 CR9C5Z 9911060 Ki = 23 nM T67363 CD7I4Y 9911639 Ki = 1.3 nM T67363 CBZ20D 9913337 IC50 = 71.5 nM T67363 CE6G5M 9914031 IC50 = 11 nM T67363 CR13IL 9914166 IC50 = 0.055 nM T67363 CQZI61 9914952 IC50 = 74 nM T67363 COT86Q 9915619 IC50 = 2.3 nM T67363 CF4J2Z 9923982 IC50 = 36 nM T67363 CUBV32 9924032 IC50 = 330 nM T67363 C8ZMX1 9929222 IC50 = 0.07 nM T67363 CJPZ87 9930471 IC50 = 1.9 nM T67363 CC42WD 9932423 IC50 = 19 nM T67363 CQ45ME 9934825 IC50 = 5.64 nM T67363 C59UEH 9934950 IC50 = 10000 nM T67363 CKRZ62 9937119 IC50 = 3 nM T67363 C0R3EL 9951932 IC50 = 0.08 nM T67363 C1UK7T 9953715 Ki = 2.5 nM T67363 C8UC3W 9953989 Ki = 45 nM T67363 CYG4S2 9954358 IC50 = 35 nM T67363 C9CKS6 9956141 IC50 = 1.18 nM T67363 C4XK2S 9956830 IC50 = 3.6 nM T67363 CDU79H 9957105 IC50 = 0.19 nM T67363 CH1Y7E 9957565 IC50 = 0.31 nM T67363 CWUC80 9958350 Ki = 2.5 nM T67363 CUIF89 9979634 IC50 = 60000 nM T67363 CT4V2Y 9979833 IC50 = 2.4 nM T67363 CIXB62 9979842 IC50 = 8.8 nM T67363 CXN45H 9983052 IC50 = 2.5 nM T67363 CYA0W2 9983143 IC50 = 2.82 nM T67363 CCR6V0 9983448 Ki = 70.9 nM T67363 CPE58N 9984136 IC50 = 0.8 nM T67363 C8NCZ4 9985786 IC50 = 0.6 nM T67363 CLB29G 9996802 IC50 > 100000 nM T67363 CP2MN7 10002412 IC50 = 1.01 nM T67363 C6CWQ8 10003119 IC50 = 11.06 nM T67363 CA2SU9 10004734 IC50 = 1.2 nM T67363 C1SHP7 10007481 IC50 = 1.7 nM T67363 CADZ52 10007574 IC50 = 0.57 nM T67363 CBT02G 10026044 IC50 = 0.8 nM T67363 CEJ31C 10027119 IC50 = 3.49 nM T67363 CGT4D2 10027594 IC50 = 233 nM T67363 C5CZ8A 10028351 IC50 = 1.9 nM T67363 C6WP7I 10028701 IC50 = 0.32 nM T67363 CY0T9L 10030149 IC50 = 3.2 nM T67363 CE2CK1 10032445 IC50 = 70 nM T67363 CGA89W 10049569 IC50 = 1 nM T67363 CD6SV4 10050710 IC50 = 80 nM T67363 CLS1F7 10051002 IC50 = 0.32 nM T67363 C5PMK2 10051658 IC50 = 1 nM T67363 COH3U6 10052945 IC50 = 0.9 nM T67363 C40FMW 10069462 IC50 = 0.2 nM T67363 C2R7TW 10069591 IC50 = 330000 nM T67363 C3WZR0 10069974 IC50 = 2.7 nM T67363 CX6H0Q 10072507 IC50 = 0.8 nM T67363 CBF7V6 10073290 IC50 = 1.24 nM T67363 CK0G2T 10073952 IC50 = 1.54 nM T67363 CC3LU6 10074467 IC50 = 1 nM T67363 CH0Y4Z 10074600 IC50 = 1.5 nM T67363 C21LFO 10076708 IC50 = 2 nM T67363 CB7R9Y 10096029 IC50 = 1.7 nM T67363 CL47PJ 10096030 IC50 = 0.83 nM T67363 CLN76R 10096459 IC50 = 0.45 nM T67363 CDEA39 10096654 IC50 = 1.9 nM T67363 C6JLQ8 10097012 IC50 = 0.32 nM T67363 CSD8L0 10097881 Ki = 0.5 nM T67363 C1YX0U 10098164 IC50 = 0.2 nM T67363 CS2A6F 10098382 IC50 = 1.18 nM T67363 CA03GD 10098780 Ki = 4 nM T67363 C1X6MY 10099012 Ki = 50 nM T67363 CDN7E3 10109428 IC50 = 6 nM T67363 C4GEW5 10111539 IC50 = 31.62 nM T67363 C58CQE 10112695 IC50 = 0.2 nM T67363 CESP84 10113832 IC50 = 9000 nM T67363 CM50IS 10116182 IC50 = 0.7 nM T67363 C9CI6R 10117329 IC50 = 37 nM T67363 CS08OY 10117330 IC50 = 37 nM T67363 CTH5X2 10118705 IC50 = 40 nM T67363 C1H4NB 10132697 IC50 = 0.6 nM T67363 C6AB5O 10132765 IC50 = 460 nM T67363 C9FN1L 10134456 IC50 = 2000 nM T67363 C5HFG7 10135509 IC50 = 0.11 nM T67363 CWT3Y7 10136986 IC50 = 3.6 nM T67363 CEO04K 10140146 IC50 = 1.1 nM T67363 COFK25 10160125 IC50 = 15 nM T67363 CNBL36 10160126 IC50 = 1800 nM T67363 CLBK65 10160411 IC50 = 14 nM T67363 CE8ZX3 10161387 IC50 = 0.4 nM T67363 C1O0GR 10162362 IC50 = 20 nM T67363 CIQ3W5 10162576 IC50 = 55 nM T67363 CX7A1Z 10164947 IC50 = 1.8 nM T67363 CDL31V 10165701 IC50 = 1.1 nM T67363 C16ZLE 10181046 IC50 = 1900 nM T67363 CV0G1X 10181237 IC50 = 0.6 nM T67363 CP64AK 10181815 IC50 = 1 nM T67363 CMNJ08 10181868 IC50 = 0.9 nM T67363 C38XFC 10182400 IC50 = 0.1 nM T67363 CXJO84 10183763 IC50 = 0.8 nM T67363 C38TOH 10184998 IC50 = 0.38 nM T67363 CO8D9C 10196873 IC50 = 2.6 nM T67363 CP26BW 10200045 IC50 = 0.93 nM T67363 C9SYN1 10201323 IC50 = 23 nM T67363 C4Z2QI 10204795 IC50 = 0.7 nM T67363 CPO60A 10208212 IC50 = 0.46 nM T67363 CBL69X 10223113 IC50 = 5 nM T67363 CPT2Q5 10224943 IC50 = 68 nM T67363 C1QN0U 10227414 IC50 = 0.5 nM T67363 C53NHL 10228662 IC50 = 9.5 nM T67363 CIZ09S 10230114 IC50 = 1.3 nM T67363 CD04YP 10240088 IC50 = 14800 nM T67363 C0M7FC 10248023 IC50 > 100000 nM T67363 C42BVA 10251325 IC50 = 0.58 nM T67363 CM9UQ8 10252576 IC50 = 1.77 nM T67363 CY8BZ3 10254053 IC50 = 1.8 nM T67363 CCV9K4 10255072 Ki = 1.6 nM T67363 C8FVA4 10255345 IC50 = 0.49 nM T67363 CHX06T 10255701 IC50 = 0.3 nM T67363 CVBS78 10256274 IC50 = 1.56 nM T67363 CUZ1I2 10256289 IC50 = 1.1 nM T67363 C73JHS 10258262 IC50 = 1.6 nM T67363 C38UIQ 10273975 IC50 = 15.85 nM T67363 C9JOB1 10274638 IC50 = 4000 nM T67363 C5YRK9 10275142 IC50 = 1.2 nM T67363 CD04QE 10279663 IC50 = 0.77 nM T67363 C7E8PX 10281105 IC50 = 110 nM T67363 CIF59V 10281222 IC50 = 53 nM T67363 C9CST0 10281487 IC50 = 0.65 nM T67363 CG4Y9X 10294880 IC50 = 200 nM T67363 CJE72C 10295656 IC50 = 116 nM T67363 C2Y9PQ 10295657 IC50 = 78 nM T67363 CR2YI9 10297636 IC50 = 1.2 nM T67363 COXW74 10320601 IC50 = 1.07 nM T67363 CH5F6W 10322871 IC50 = 75 nM T67363 CUZ8V6 10323749 IC50 = 7 nM T67363 CXMC15 10325138 IC50 = 7 nM T67363 CM0X6T 10325997 Ki = 0.7 nM T67363 CX52DZ 10338161 IC50 = 1900 nM T67363 C84KLV 10340994 IC50 = 51 nM T67363 CKA8S0 10343706 IC50 = 0.39 nM T67363 CYXW23 10343956 IC50 = 56000 nM T67363 CN7B1W 10344154 IC50 = 0.25 nM T67363 CR5VI0 10344187 IC50 = 0.7 nM T67363 CD1C7I 10345263 IC50 = 2.1 nM T67363 CF18LZ 10345912 IC50 = 1490 nM T67363 CTS1H5 10346321 IC50 = 0.31 nM T67363 C62KDF 10347784 IC50 > 10000 nM T67363 C1ZC2P 10348465 IC50 = 0.08 nM T67363 CI3AF9 10367229 IC50 = 28.1 nM T67363 CXF75S 10367371 IC50 = 1.22 nM T67363 CQ04DG 10367832 IC50 = 0.75 nM T67363 CY1R0K 10368440 IC50 = 142 nM T67363 CL3RB6 10368999 IC50 = 0.6 nM T67363 CVOY03 10369856 IC50 = 31 nM T67363 CQ4H3K 10386147 IC50 = 1.7 nM T67363 C5CMH6 10391088 IC50 = 3 nM T67363 C31WGJ 10391128 IC50 = 0.7 nM T67363 C8D9QH 10391556 IC50 = 1.26 nM T67363 C8PNS3 10391689 IC50 = 2.6 nM T67363 CC0L8M 10392074 IC50 = 8 nM T67363 CB56UW 10392450 IC50 = 1.8 nM T67363 CEQC07 10392868 IC50 = 2 nM T67363 C4H3JG 10393220 IC50 = 0.3 nM T67363 C1ZM6J 10393879 IC50 = 5 nM T67363 CH4R7P 10394263 IC50 = 6.4 nM T67363 CL9SM7 10404377 IC50 > 100000 nM T67363 CEP9G0 10410948 IC50 = 2.8 nM T67363 CX1D5C 10411516 IC50 = 1 nM T67363 CO0FY6 10411523 IC50 = 281 nM T67363 CXZT32 10411746 IC50 = 22.3 nM T67363 CB3K1N 10412117 IC50 = 0.44 nM T67363 C7B3MO 10412184 IC50 = 1.2 nM T67363 CR0F1T 10412890 IC50 = 0.8 nM T67363 C7NQW0 10413380 IC50 = 20.6 nM T67363 CFP6E5 10414330 IC50 > 100000 nM T67363 C6HUB8 10414462 IC50 = 0.8 nM T67363 C3PI8C 10414569 IC50 = 3.73 nM T67363 C8UZE4 10415159 IC50 = 0.4 nM T67363 CZ12CP 10415384 IC50 = 2 nM T67363 C3K6LV 10415627 IC50 = 0.2 nM T67363 C5VN6I 10427709 IC50 > 100000 nM T67363 CZF8I1 10432418 IC50 = 3 nM T67363 CUHY62 10433896 IC50 = 0.4 nM T67363 CRP82B 10435346 IC50 = 64 nM T67363 C9F2QA 10436174 IC50 = 1.77 nM T67363 C1ME0S 10436235 IC50 = 2.7 nM T67363 C1IFC6 10436829 IC50 = 0.3 nM T67363 C04HQK 10437073 IC50 = 1.5 nM T67363 C1EH5P 10439474 IC50 = 331.8 nM T67363 C0IA8K 10455265 IC50 = 147000 nM T67363 C1XTA5 10456473 IC50 = 0.35 nM T67363 C6G9YM 10457584 IC50 = 1 nM T67363 C9ZN4U 10457840 IC50 = 1.1 nM T67363 CX69EL 10458074 Ki = 56000 nM T67363 C6P0ZM 10458809 IC50 = 49 nM T67363 CQV26D 10459311 IC50 > 100000 nM T67363 CTZC60 10461016 IC50 > 100000 nM T67363 CA27PJ 10478285 IC50 = 0.9 nM T67363 C8EKH9 10479033 IC50 = 1.23 nM T67363 C5FX7L 10479186 IC50 = 3.81 nM T67363 C0NVB7 10479802 IC50 = 2.17 nM T67363 COJW10 10480848 Ki = 0.7 nM T67363 CT04RE 10481345 IC50 = 0.29 nM T67363 C6IAB4 10482388 IC50 = 2.09 nM T67363 C9OM3L 10482416 IC50 = 0.9 nM T67363 C45MRF 10483616 IC50 = 44 nM T67363 CM0ZW9 10503055 IC50 > 100000 nM T67363 C1U8TQ 10504200 IC50 = 40 nM T67363 CF24JN 10505627 IC50 = 360 nM T67363 CR26WA 10506313 IC50 = 7.1 nM T67363 C3W8VJ 10507104 IC50 = 13 nM T67363 CZ70VF 10507218 IC50 = 120 nM T67363 CC58KL 10507483 IC50 > 1000 nM T67363 CXS79H 10507484 IC50 > 1000 nM T67363 CW37AZ 10526036 IC50 = 2 nM T67363 C7DQU0 10526203 Ki = 1100 nM T67363 CD6T3L 10527653 IC50 = 1 nM T67363 C0T5IM 10529317 IC50 > 1000 nM T67363 CM4Z9C 10529546 IC50 = 74 nM T67363 CUJ3S8 10529815 IC50 > 1000 nM T67363 CUY9Q0 10529865 IC50 = 300 nM T67363 C61HVA 10530613 IC50 = 10 nM T67363 C2L1PJ 10531967 IC50 = 4.6 nM T67363 CBS2F4 10548981 IC50 = 160 nM T67363 C8Y3PH 10551831 IC50 > 100000 nM T67363 CEO2N5 10552647 IC50 = 10.6 nM T67363 C7BLP8 10553605 IC50 = 46 nM T67363 CZD20R 10555279 IC50 = 8.8 nM T67363 CAWF40 10574237 Ki = 9200 nM T67363 C75XGA 10574888 IC50 = 125000 nM T67363 C73VFG 10574923 IC50 > 100000 nM T67363 C9TO2C 10577800 IC50 > 1000 nM T67363 CQ96ZW 10578645 IC50 > 1000 nM T67363 CU75WP 10578810 IC50 = 4.7 nM T67363 C0U1CG 10582643 IC50 = 27 nM T67363 CDK10F 10597871 IC50 > 100000 nM T67363 CC52PM 10601502 IC50 > 100000 nM T67363 CP0O3V 10601903 IC50 > 1000 nM T67363 C39IPX 10603319 IC50 = 8.5 nM T67363 CPVM74 10604005 IC50 > 100000 nM T67363 CDXB14 10606654 IC50 = 1 nM T67363 C7N8UQ 10621705 IC50 = 0.9 nM T67363 C35QBJ 10623736 IC50 > 100000 nM T67363 C4V9FB 10626190 IC50 > 1000 nM T67363 CUBJ20 10628601 IC50 = 52 nM T67363 C1TKQ4 10645607 IC50 = 160 nM T67363 CMB93Z 10645847 Ki = 4200 nM T67363 CS5PN3 10647720 IC50 = 2 nM T67363 CM54PX 10647971 IC50 = 3 nM T67363 C5ABX8 10648597 Ki = 510 nM T67363 CX98VN 10648960 IC50 = 73 nM T67363 CY38BT 10649923 IC50 = 54 nM T67363 CHV18W 10650104 IC50 = 10 nM T67363 CW5KO9 10650595 IC50 = 840 nM T67363 C4QO9H 10651012 IC50 = 35 nM T67363 C6I7GM 10673034 IC50 > 1000 nM T67363 C5C4KF 10673305 IC50 = 44 nM T67363 C1K4VA 10673587 IC50 = 120 nM T67363 CNZ52W 10674738 IC50 = 52 nM T67363 CY10JG 10678157 IC50 = 37 nM T67363 CMV21P 10678163 IC50 = 1 nM T67363 C6R4MV 10678165 IC50 = 20000 nM T67363 C6U0EH 10691302 IC50 = 23 nM T67363 CM4I0K 10692763 Ki = 15 nM T67363 C6G5SF 10696089 IC50 > 100000 nM T67363 C3SF8N 10697605 IC50 = 34 nM T67363 CFG8O6 10698251 IC50 = 150 nM T67363 CYV8S2 10698274 IC50 = 28 nM T67363 C9GTM8 10713257 IC50 > 1000 nM T67363 CIMF59 10715577 Ki = 1150 nM T67363 C3CG9M 10717156 IC50 = 100000 nM T67363 CY40LK 10720760 IC50 = 15 nM T67363 CA4HQ9 10721455 IC50 < 0.1 nM T67363 CYM68T 10721510 IC50 = 70 nM T67363 CMW37K 10737695 IC50 > 1000 nM T67363 CMCP54 10737883 IC50 > 100000 nM T67363 C0WB5V 10741543 IC50 > 100000 nM T67363 CQ43HK 10743381 IC50 > 100000 nM T67363 CPD32M 10744420 IC50 > 1000 nM T67363 CPW19S 10744934 IC50 = 170 nM T67363 CS7YL2 10745179 IC50 = 18 nM T67363 C5N0JC 10745304 IC50 = 290 nM T67363 CPQ9N3 10746038 IC50 > 100000 nM T67363 CTZG52 10746372 IC50 = 4.9 nM T67363 C65WOR 10766035 IC50 = 2 nM T67363 C4XFU2 10767331 IC50 = 3 nM T67363 CO15MH 10769104 IC50 = 240 nM T67363 CDZM40 10781802 IC50 > 100000 nM T67363 CR2Y3H 10788405 Ki = 1000 nM T67363 CB83FZ 10789670 IC50 = 1.8 nM T67363 CRLY08 10790058 IC50 = 26 nM T67363 CGI2S3 10792202 IC50 = 16 nM T67363 CKU3Z4 10792272 IC50 = 51 nM T67363 C03KUV 10792275 IC50 > 1000 nM T67363 C90EQR 10793103 IC50 = 56 nM T67363 C7X1ZK 10793322 IC50 > 1000 nM T67363 C9L4KF 10793351 IC50 = 10 nM T67363 CQSR19 10814133 IC50 = 0.08 nM T67363 CB68AD 10814586 IC50 > 1000 nM T67363 CXQD50 10814626 IC50 > 100000 nM T67363 CD3P4W 10815546 IC50 > 1000 nM T67363 CNG0H1 10816131 IC50 > 1000 nM T67363 CI7HF0 10830837 IC50 > 1000 nM T67363 CT41YH 10831740 IC50 = 7200 nM T67363 CCW4P0 10838744 IC50 = 81 nM T67363 CQ7SB0 10839335 IC50 = 460 nM T67363 C06QAI 10839976 IC50 = 170 nM T67363 CTJ61U 10840969 IC50 = 360 nM T67363 C7EB4Y 10844291 IC50 = 4 nM T67363 C9XK7J 10844292 IC50 = 6 nM T67363 CX09YP 10906526 IC50 = 141 nM T67363 CIV0X1 10961560 IC50 = 39 nM T67363 C08BCF 10993678 IC50 = 13 nM T67363 CDK7W9 10994476 IC50 = 53 nM T67363 C3W9NV 11039087 IC50 = 2.4 nM T67363 CTW0P5 11102917 IC50 = 14 nM T67363 C4U5OQ 11122429 IC50 = 0.25 nM T67363 C79OJR 11133736 IC50 = 53 nM T67363 C36HWS 11134241 IC50 = 0.35 nM T67363 CU8FZ2 11146108 IC50 = 3.6 nM T67363 C3S5VP 11157853 Ki = 2.27 nM T67363 CM98TK 11165725 IC50 = 0.21 nM T67363 CJU1K7 11200734 IC50 = 0.16 nM T67363 C4HFS8 11234619 IC50 > 50000 nM T67363 CDN62X 11269177 IC50 > 50000 nM T67363 CK07JV 11292789 IC50 = 0.52 nM T67363 CNZ17L 11330668 Ki = 6.3 nM T67363 CZO3H7 11399588 IC50 = 16 nM T67363 C9L2OX 11452690 IC50 = 0.24 nM T67363 CC4S7U 11486328 IC50 = 0.65 nM T67363 CDIR54 11486773 IC50 = 0.24 nM T67363 CX9G5B 11534748 IC50 = 38 nM T67363 C5NEM0 11546965 IC50 = 0.6 nM T67363 CFZ2O9 11613998 IC50 = 16000 nM T67363 C8SC4J 11628511 IC50 = 2.07 nM T67363 CDV02G 11628719 IC50 = 6500 nM T67363 CWU71P 11699824 IC50 = 9 nM T67363 CGU84F 11721315 IC50 = 880 nM T67363 C2ONX6 11721442 IC50 = 36 nM T67363 CJ63KS 11733125 IC50 = 3 nM T67363 CS1Q9P 11744536 IC50 = 0.94 nM T67363 CZ2C3R 11753914 IC50 = 0.13 nM T67363 CJ3Q2G 11754575 IC50 = 1.2 nM T67363 C25GTJ 11756112 IC50 = 3.54 nM T67363 CPXI40 11757187 IC50 = 0.2 nM T67363 C3DCM0 11757316 IC50 = 1.6 nM T67363 CEN37T 11757623 IC50 = 48 nM T67363 CG26EJ 11762165 Ki = 20 nM T67363 C2L3HF 11797838 IC50 = 6 nM T67363 C5GTQ0 11798113 IC50 > 100000 nM T67363 CFL9C4 11799328 IC50 = 106 nM T67363 C4U1TD 11800065 IC50 = 26 nM T67363 CZ06CB 11800170 IC50 = 62 nM T67363 CD0GH5 11800573 IC50 = 160 nM T67363 COT19X 11800615 IC50 = 26 nM T67363 CYC1X9 11800819 IC50 = 600 nM T67363 CR2CL6 11842612 IC50 = 0.96 nM T67363 CF8YK0 11965389 IC50 = 0.5 nM T67363 CW7T9U 11965462 IC50 = 4.4 nM T67363 CSPA57 12071479 Ki = 550 nM T67363 C1E9BA 12096120 IC50 = 0.058 nM T67363 CFRW03 12135085 Ki = 5.1 nM T67363 CZTJ02 12795460 IC50 = 40.9 nM T67363 C04GKV 15030977 IC50 > 300000 nM T67363 C3KUC7 15462235 IC50 = 0.3 nM T67363 CMES74 15486068 Ki = 1.9 nM T67363 C2YG3M 15491369 Ki = 280 nM T67363 COEP73 15491370 Ki = 33 nM T67363 CZ2R8G 15491452 IC50 = 15 nM T67363 CN0LX5 15491453 IC50 = 11 nM T67363 C3VOW7 15491454 IC50 = 12 nM T67363 CZX58V 15516067 Ki = 22000 nM T67363 CDVB07 15850631 IC50 = 3 nM T67363 CG9FV3 15850632 IC50 = 10 nM T67363 CM8G3S 15859412 IC50 = 9 nM T67363 CW8LN2 15859413 IC50 = 41 nM T67363 CT1DI8 15859414 IC50 = 10 nM T67363 C95OGC 15859418 IC50 = 2 nM T67363 CEC41O 15859419 IC50 = 4 nM T67363 CFJ08N 15859420 IC50 = 3 nM T67363 CUQ9A2 15859421 IC50 = 2 nM T67363 C56IZT 15859422 IC50 = 3 nM T67363 CE6FO4 15859423 IC50 = 16 nM T67363 C1VMK9 15859424 IC50 = 1100 nM T67363 C8QIB4 15888084 Ki = 8 nM T67363 CDUW15 16088010 IC50 = 2150 nM T67363 CR6ZY3 16088011 IC50 = 34.4 nM T67363 C4ZW7G 16115221 IC50 = 304 nM T67363 CW41XZ 16663331 IC50 = 110 nM T67363 CDUC32 16665100 IC50 = 703 nM T67363 CTGC60 16678135 IC50 = 84 nM T67363 C4T7ZE 16724119 IC50 = 20 nM T67363 CV14TI 16739275 IC50 = 26 nM T67363 CU8YQ3 16756502 IC50 = 2.4 nM T67363 CJUK37 16756504 IC50 = 140 nM T67363 C0KW3V 16756505 IC50 = 1200 nM T67363 C04JOX 16756621 IC50 = 3400 nM T67363 C4CU7T 16756622 IC50 = 3300 nM T67363 CFH96E 16756623 IC50 = 690 nM T67363 CXK79J 16756847 IC50 = 21 nM T67363 CB15RX 16756849 IC50 = 6.3 nM T67363 CM18ZN 16756955 IC50 = 1600 nM T67363 CL38IU 16756956 IC50 = 4 nM T67363 CW5P8L 16756957 IC50 = 980 nM T67363 C78CUA 18322736 IC50 = 0.3 nM T67363 CG67XJ 18346107 IC50 = 71.7 nM T67363 C4VFQ1 18346108 IC50 = 18.1 nM T67363 CX30NF 18346110 IC50 = 34.5 nM T67363 C2DN9B 18394355 Ki = 110 nM T67363 C8Z3NC 18394360 Ki = 5 nM T67363 C9B2VL 18394361 Ki = 3.5 nM T67363 CAOR56 18660413 IC50 = 240 nM T67363 CE3F1W 18768256 IC50 = 210 nM T67363 C0O6XT 19076730 IC50 = 19 nM T67363 CXLO94 20587795 IC50 = 4 nM T67363 CW64DV 20666951 IC50 = 4760 nM T67363 C85SOV 20666970 IC50 = 3.2 nM T67363 C61WDP 20666971 IC50 = 19.1 nM T67363 CX52NV 20666990 IC50 = 2.6 nM T67363 CVJ8N2 20667011 IC50 = 1.1 nM T67363 CMV17G 20667012 IC50 = 24 nM T67363 CQ8ME6 20667015 IC50 = 0.8 nM T67363 CX1NI3 20691527 IC50 = 10.9 nM T67363 C6VZA8 20709789 IC50 = 150 nM T67363 C6V9FP 20817441 IC50 = 2700 nM T67363 CTH25W 20950504 EC50 = 1.6 nM T67363 CEI27V 21053920 IC50 > 10000 nM T67363 C3TR2D 21191396 IC50 = 2.9 nM T67363 CE5Z3R 21191398 IC50 = 9 nM T67363 CGI19E 21191399 IC50 = 2.5 nM T67363 CN1Q0M 21191405 IC50 = 0.16 nM T67363 C3GK7N 21191409 IC50 = 21 nM T67363 CQJ5Z3 21191417 IC50 = 5.6 nM T67363 CU4FN2 21191441 IC50 = 6.1 nM T67363 CM96YE 21191461 IC50 = 0.27 nM T67363 C7XYV3 21191470 IC50 = 0.11 nM T67363 CUJS70 21699778 IC50 = 48 nM T67363 C2N6QA 21927945 IC50 = 12 nM T67363 C19UCA 21934501 IC50 = 0.61 nM T67363 CB53QY 21955393 IC50 = 500 nM T67363 CI0UK9 21955407 IC50 = 1000 nM T67363 CT0NH1 21955413 IC50 = 220 nM T67363 CV0E3C 21955419 IC50 = 23 nM T67363 CU1RF9 21955424 IC50 = 200 nM T67363 CX84CU 21955425 IC50 = 620 nM T67363 CY7UQ0 21955428 IC50 = 100 nM T67363 CACY12 21955467 IC50 = 5000 nM T67363 CCJT57 21955505 IC50 = 10000 nM T67363 C7JIA3 21967988 IC50 = 4.7 nM T67363 C7EW4N 21967992 IC50 = 11.2 nM T67363 C7WPF4 21967993 IC50 = 6.1 nM T67363 C3B4WA 21967994 IC50 = 21.3 nM T67363 CZG18W 21967995 IC50 = 49.8 nM T67363 CH78QV 21967996 IC50 = 51.6 nM T67363 CR7O8I 21982386 Ki = 280 nM T67363 CE4L1Y 21982428 Ki = 30 nM T67363 CFJ3N2 21982435 Ki = 4 nM T67363 C5I6GE 21982524 Ki = 100 nM T67363 C8TX5F 22092675 Ki > 10000 nM T67363 C2MZ9G 22092797 Ki = 350 nM T67363 C2L7HP 22092801 Ki = 360 nM T67363 CZNA37 22092805 Ki = 60 nM T67363 C2VAY9 22092806 Ki = 14 nM T67363 CL2V5Y 22092807 Ki = 25 nM T67363 CM5J8B 22092817 Ki = 4 nM T67363 C34TEM 22092820 Ki = 180 nM T67363 CUZ34O 22092829 Ki = 220 nM T67363 CMCY21 22092833 Ki = 700 nM T67363 CG41IR 22092922 Ki = 1.4 nM T67363 CZYF73 22092924 Ki = 60 nM T67363 C6XG1K 22092927 Ki = 300 nM T67363 CW31ES 22092931 Ki = 20 nM T67363 C7ISM4 22092936 Ki = 90 nM T67363 C1KVO9 22092956 Ki > 10000 nM T67363 CT6N9S 22094645 IC50 = 0.77 nM T67363 CMS31G 22098946 IC50 = 3 nM T67363 CE5G2I 22098949 IC50 = 21 nM T67363 C2U1YQ 22098952 IC50 = 4.9 nM T67363 CEU65M 22098953 IC50 = 155 nM T67363 CO4JK1 22098959 IC50 = 5.7 nM T67363 CN1Q2O 22098975 IC50 = 0.45 nM T67363 C94AUL 22098977 IC50 = 7.1 nM T67363 CM0JY3 22319462 IC50 = 7 nM T67363 C7W3XI 22347498 IC50 = 1000 nM T67363 C7T5LS 22347500 IC50 = 525 nM T67363 CGR8U4 22347512 IC50 = 1.5 nM T67363 CHP6U7 22347519 IC50 = 0.4 nM T67363 CJ03SP 22347541 IC50 = 36 nM T67363 CE2G6D 22347593 IC50 = 0.9 nM T67363 CIO36K 22347604 IC50 = 1.7 nM T67363 CA2C8K 22347617 IC50 = 776 nM T67363 C5K8AO 22347633 IC50 = 2 nM T67363 CLTQ62 22591754 Ki = 11.1 nM T67363 CVT3D0 22591800 Ki = 10.4 nM T67363 C40HYI 22591827 Ki = 1.4 nM T67363 CD72KM 22591867 Ki = 16.6 nM T67363 CXVB03 22594242 IC50 = 0.3 nM T67363 CDJH42 22594251 IC50 = 0.3 nM T67363 CPF73W 22594331 IC50 = 45 nM T67363 CHR03I 22594351 IC50 = 584 nM T67363 CFL7X5 22594355 IC50 = 842 nM T67363 CZ9NX2 22678222 IC50 = 0.82 nM T67363 C9YZU3 22678243 IC50 = 0.72 nM T67363 CMET78 23435760 IC50 > 100000 nM T67363 CKF08G 23435786 IC50 > 100000 nM T67363 CX6AR9 23627460 IC50 = 790 nM T67363 CYND24 23729562 IC50 = 2730 nM T67363 C96PUZ 23729563 IC50 = 12200 nM T67363 CZ17YE 23731146 IC50 = 103 nM T67363 CHXT18 23731243 IC50 = 490 nM T67363 CEA9Z8 23731244 IC50 = 770 nM T67363 CNK5O6 23731245 IC50 = 1200 nM T67363 C6W9OS 23731246 IC50 = 1300 nM T67363 CK7OW6 24779699 Ki = 0.5 nM T67363 CR72IF 24864718 IC50 = 2600 nM T67363 C9L0QD 24864721 IC50 = 1 nM T67363 CXH2G0 24864898 IC50 = 7 nM T67363 C7TPO5 24865624 IC50 = 290 nM T67363 C5DVB6 24865625 IC50 = 600 nM T67363 C8G2FE 24866358 IC50 = 440 nM T67363 C6I1OF 24866515 IC50 = 280 nM T67363 CZ7QL8 24866516 IC50 = 400 nM T67363 CNCH18 24866519 IC50 = 520 nM T67363 CY6WR2 24872066 IC50 = 642 nM T67363 CUM4E3 24872070 IC50 = 1050 nM T67363 CG09DH 24872646 IC50 = 239 nM T67363 CRS65Q 24873110 IC50 = 648 nM T67363 C0HZ7E 24873345 IC50 = 402 nM T67363 C28KAH 24873465 IC50 = 38 nM T67363 C1PB6T 25025343 IC50 = 2900 nM T67363 CDA2B9 25025730 IC50 = 200 nM T67363 CD2L7Z 25025937 IC50 = 130 nM T67363 CIS68P 25032865 IC50 = 0.7 nM T67363 CB6H7T 25107570 IC50 > 100000 nM T67363 CC40FO 25107571 IC50 > 100000 nM T67363 C1QC4Y 25107572 IC50 > 100000 nM T67363 C84XCZ 25107635 IC50 > 100000 nM T67363 CRV78W 25107708 IC50 > 100000 nM T67363 C3V7JU 25107773 IC50 > 100000 nM T67363 C43TCR 25183860 IC50 = 830 nM T67363 CR92LD 25184415 IC50 = 960 nM T67363 CC4A5X 25194118 IC50 = 73.28 nM T67363 CK73JX 25194121 IC50 = 10.8 nM T67363 C3J7GQ 28510125 IC50 > 1000 nM T67363 CLX6T9 28510811 IC50 = 9.5 nM T67363 CM37RS 42607047 IC50 = 16 nM T67363 C7K4HE 42607050 IC50 = 5.4 nM T67363 CSK94Y 44266085 IC50 = 16.5 nM T67363 CF2MV4 44266092 IC50 = 0.7 nM T67363 C9UP0S 44266099 IC50 = 36.7 nM T67363 C5FS2W 44266101 IC50 = 2.3 nM T67363 C28BEI 44266148 IC50 = 0.6 nM T67363 CC1Y0A 44266157 IC50 = 0.3 nM T67363 C37XYK 44266161 IC50 = 0.4 nM T67363 C3BKQ7 44266189 IC50 = 0.3 nM T67363 CQK2N1 44266208 IC50 = 0.9 nM T67363 CL4GY7 44266216 IC50 = 0.9 nM T67363 CD4FP1 44266861 Ki = 70 nM T67363 C80HOG 44266865 Ki = 170 nM T67363 CCE98M 44266878 Ki = 1700 nM T67363 CMP67S 44266882 Ki = 60 nM T67363 CSJ2H3 44266883 Ki = 80 nM T67363 CGEZ18 44266884 Ki = 8 nM T67363 C0AFL5 44266888 Ki = 75 nM T67363 CN29ZD 44266890 Ki = 300 nM T67363 CQ5A0G 44266898 Ki = 560 nM T67363 CB9Y6U 44266900 Ki > 10000 nM T67363 C5Z0IM 44266901 Ki = 500 nM T67363 C0JD8S 44266906 Ki = 80 nM T67363 CNT0G1 44266907 Ki = 1 nM T67363 CM7TD3 44266908 Ki = 20 nM T67363 C1PKT0 44266909 Ki = 100 nM T67363 C17DPA 44266910 Ki = 74 nM T67363 CJ5TO6 44266911 Ki = 300 nM T67363 CHD76I 44266913 Ki = 4 nM T67363 CU3D7W 44266915 Ki = 1000 nM T67363 CE2B5X 44266916 Ki > 10000 nM T67363 CIJ0A1 44266919 Ki = 10 nM T67363 C23SWQ 44266924 Ki = 14 nM T67363 CD4AK8 44266927 Ki = 800 nM T67363 C3G7WH 44266952 Ki = 750 nM T67363 CV9MK7 44266954 Ki = 120 nM T67363 C2RIE4 44266963 Ki > 10000 nM T67363 C3IE6Z 44266969 Ki = 900 nM T67363 C4XE6G 44266974 Ki = 210 nM T67363 CX7S1E 44266978 Ki = 850 nM T67363 CPV4N0 44266984 Ki = 800 nM T67363 C3PED5 44266985 Ki = 160 nM T67363 CPS49K 44267000 Ki > 10000 nM T67363 CKY6J1 44267010 Ki = 11 nM T67363 CNM1H2 44267012 Ki = 100 nM T67363 CP7NK3 44267015 Ki > 10000 nM T67363 C2E8YZ 44273729 Ki = 10 nM T67363 CUV4A7 44277982 IC50 = 3.1 nM T67363 C03OEI 44277984 IC50 = 10000 nM T67363 CMGY79 44277986 IC50 = 144 nM T67363 CL36QJ 44278084 IC50 = 8.9 nM T67363 CFV24Z 44278300 IC50 = 2330 nM T67363 C9RJY3 44278338 IC50 = 100 nM T67363 C9DE0N 44278380 IC50 = 0.5 nM T67363 CU12EY 44278381 IC50 = 16 nM T67363 CATY17 44278385 IC50 = 50.5 nM T67363 CN2FA3 44278391 IC50 = 14 nM T67363 COI3M9 44278397 IC50 = 0.1 nM T67363 CD8E2K 44278410 IC50 = 3.8 nM T67363 COD26Y 44278417 IC50 = 0.9 nM T67363 C34VTL 44278469 IC50 = 1.5 nM T67363 CHR9D4 44278470 IC50 = 0.3 nM T67363 CJC7G4 44278548 IC50 = 1000 nM T67363 CL9FU4 44278570 IC50 = 311 nM T67363 CQ7B4A 44278586 IC50 = 1000 nM T67363 C7VI1M 44278647 IC50 = 0.2 nM T67363 CL36VA 44278649 IC50 = 72 nM T67363 CN03LX 44278749 IC50 = 5000 nM T67363 C2PN5A 44278774 IC50 = 1000 nM T67363 C6Q4ZP 44278906 IC50 = 88.2 nM T67363 C8VDT0 44278907 IC50 = 43.5 nM T67363 C48KBZ 44283063 IC50 = 4 nM T67363 CF7C8I 44283067 IC50 = 0.63 nM T67363 C2FV0E 44283118 IC50 = 1830 nM T67363 CK0RD4 44283161 IC50 = 10.3 nM T67363 CXE01A 44283190 IC50 = 3 nM T67363 C12RPS 44283197 IC50 = 0.48 nM T67363 C4VW3I 44283198 IC50 = 0.46 nM T67363 C9ZQW4 44283202 IC50 = 3.5 nM T67363 C6KLR5 44283203 IC50 = 10.6 nM T67363 CMV19L 44283204 IC50 = 23 nM T67363 CNI3F9 44283232 IC50 = 32 nM T67363 C74CWT 44283235 IC50 = 0.2 nM T67363 CN45TM 44283254 IC50 = 9.7 nM T67363 CVS5P4 44283263 IC50 = 3.8 nM T67363 CX2PH8 44283275 IC50 = 19.4 nM T67363 CH29QO 44283299 IC50 = 122 nM T67363 C7FCI9 44283300 IC50 = 1.2 nM T67363 C2M4JN 44283364 IC50 = 1.8 nM T67363 C5R6PO 44283380 IC50 = 0.49 nM T67363 C2XCB4 44283544 Ki = 7 nM T67363 C09EHM 44283639 IC50 = 2.2 nM T67363 C50ETI 44283738 Ki = 170 nM T67363 C2C5SF 44283748 Ki = 12 nM T67363 C4MS2Q 44291130 IC50 = 15 nM T67363 CNFY65 44291131 IC50 = 0.4 nM T67363 C5V1GK 44291221 IC50 = 1000 nM T67363 CGAP28 44291486 IC50 = 10 nM T67363 CEQC79 44291493 IC50 = 1.3 nM T67363 C2XQ4L 44291498 IC50 = 36 nM T67363 CUZ73G 44291499 IC50 = 1.3 nM T67363 CYBC46 44291535 IC50 = 5000 nM T67363 C3D5RJ 44291564 IC50 = 1 nM T67363 CZPG92 44291580 IC50 = 61.2 nM T67363 CGI6P2 44291581 IC50 = 5000 nM T67363 CTF48H 44291622 IC50 = 10 nM T67363 CT7XR9 44291632 IC50 = 3.6 nM T67363 C0YFB7 44291633 IC50 = 5000 nM T67363 CFI75J 44291642 IC50 = 5000 nM T67363 C9DLN5 44291646 IC50 = 5000 nM T67363 C35UPE 44291659 IC50 = 9.4 nM T67363 CC5N1G 44291660 IC50 = 500 nM T67363 CTXY96 44291661 IC50 = 103 nM T67363 CQ4UT5 44291686 IC50 = 11.6 nM T67363 CDCQ13 44291687 IC50 = 1000 nM T67363 CTI9X0 44291689 IC50 = 50000 nM T67363 C28SEF 44291690 IC50 = 10000 nM T67363 C1QU9G 44291691 IC50 = 39 nM T67363 C5V2SN 44291727 IC50 = 1000 nM T67363 C10EFC 44291749 IC50 = 3 nM T67363 CU9J0T 44291822 IC50 = 50000 nM T67363 C6V7EZ 44291823 IC50 = 5000 nM T67363 CAN87S 44291860 IC50 = 17.6 nM T67363 COE2X4 44291861 IC50 = 1000 nM T67363 CTN76I 44291917 IC50 = 50000 nM T67363 CHY7U6 44291921 IC50 = 76 nM T67363 CQN4U3 44291938 IC50 = 15.5 nM T67363 CL54WA 44291970 IC50 = 500 nM T67363 C3G5AD 44291971 IC50 = 5000 nM T67363 C6IX7F 44291999 IC50 = 1.5 nM T67363 CF6WA7 44292000 IC50 = 1.5 nM T67363 CHC8S4 44292029 IC50 = 17 nM T67363 CX9Z4D 44292030 IC50 = 46.6 nM T67363 C09ARF 44292034 IC50 = 19 nM T67363 C5B0FW 44292129 IC50 = 82 nM T67363 C1PVF7 44292130 IC50 = 48 nM T67363 CKO64J 44292131 IC50 = 4.2 nM T67363 CDBH98 44292356 IC50 = 130 nM T67363 C0EV2X 44292357 IC50 = 1 nM T67363 CD91SB 44296029 Ki = 490 nM T67363 CESC21 44296030 Ki = 2 nM T67363 C0NBT5 44296032 Ki = 1.5 nM T67363 C0EIC6 44296106 Ki = 150 nM T67363 CDX37F 44296107 Ki = 85 nM T67363 CXM37J 44296126 Ki = 9 nM T67363 CBY2N4 44296179 Ki = 2 nM T67363 C1BDP7 44296242 Ki = 8000 nM T67363 C0R6QX 44296243 Ki = 35 nM T67363 CYA4E9 44296248 Ki = 28 nM T67363 CAFV23 44296408 IC50 = 0.2 nM T67363 C74ZEK 44296431 IC50 = 0.2 nM T67363 CFN8Q6 44296449 Ki = 11 nM T67363 C1YD3S 44296450 Ki = 3000 nM T67363 CYSG84 44296458 IC50 = 0.3 nM T67363 C4FI2N 44296514 IC50 = 9 nM T67363 C9U3QW 44296519 IC50 = 0.2 nM T67363 CQHJ16 44296532 IC50 = 1 nM T67363 CX0Q1T 44296543 Ki = 1250 nM T67363 C2TE9R 44296548 IC50 = 1.4 nM T67363 C5GY7H 44296579 IC50 = 1.1 nM T67363 CYZT93 44296580 IC50 = 1.9 nM T67363 C7S1JY 44296604 IC50 = 0.8 nM T67363 CP89DV 44296642 IC50 = 1.4 nM T67363 C1KYA3 44296682 IC50 = 3000 nM T67363 CH0JP8 44296684 IC50 = 570 nM T67363 CC0TN6 44296689 IC50 = 15000 nM T67363 CUEC26 44296697 IC50 = 760 nM T67363 C2NU5B 44296726 IC50 = 350 nM T67363 CZ17IX 44296740 IC50 = 112 nM T67363 C3A7PY 44296742 IC50 = 5000 nM T67363 CAH14O 44296744 IC50 = 200 nM T67363 CZG93V 44296762 IC50 = 20 nM T67363 CJRK46 44296797 IC50 = 1660 nM T67363 CY26ES 44296824 IC50 = 1.4 nM T67363 CCEF03 44296851 IC50 = 0.2 nM T67363 C27UPR 44296852 IC50 = 0.7 nM T67363 C0FK5Q 44296857 IC50 = 2.7 nM T67363 CR9U6E 44296858 IC50 = 9.3 nM T67363 CS2E4W 44296864 IC50 = 580 nM T67363 CS62KL 44296866 IC50 = 15000 nM T67363 C0KY3B 44296868 IC50 = 40 nM T67363 C27HKT 44296892 IC50 = 200 nM T67363 CVAF21 44296901 IC50 = 2.1 nM T67363 C5O8IC 44296903 IC50 = 21 nM T67363 CTFP95 44297069 IC50 = 246 nM T67363 CJSM48 44300960 IC50 = 130 nM T67363 CFID68 44300972 IC50 = 7 nM T67363 CX2PK9 44300973 IC50 = 0.3 nM T67363 CA78QS 44300974 IC50 = 48 nM T67363 CB1E5I 44300977 IC50 = 140 nM T67363 CPJU95 44300981 IC50 = 42 nM T67363 CH8V3S 44300983 IC50 = 1400 nM T67363 CSCA61 44301010 IC50 = 37 nM T67363 C7SM9X 44301064 IC50 = 15 nM T67363 CWP52F 44301068 IC50 = 6 nM T67363 C7Q0SU 44301082 IC50 = 35 nM T67363 CLCO73 44301083 IC50 = 7 nM T67363 CC4LO8 44301244 IC50 = 3 nM T67363 C7VC5T 44301286 IC50 = 9 nM T67363 CI39XL 44301310 IC50 = 22 nM T67363 CZ14EM 44301350 IC50 = 80 nM T67363 C9QIP0 44303539 IC50 = 5 nM T67363 CC3H4P 44303550 IC50 = 4 nM T67363 C39FGB 44303551 IC50 = 5 nM T67363 CA3X5V 44303563 IC50 = 2 nM T67363 C4AO7I 44303592 IC50 = 2 nM T67363 CPX4L1 44303611 IC50 = 3 nM T67363 CRJP53 44303836 IC50 = 2 nM T67363 CTBK03 44303837 IC50 = 2 nM T67363 CUEQ19 44305411 Ki = 1500 nM T67363 C1ZQV9 44305412 Ki = 13 nM T67363 CLA5T4 44305517 Ki = 30 nM T67363 C3QI7K 44305536 Ki = 2000 nM T67363 CS5ND4 44305600 Ki = 2000 nM T67363 CP41LN 44305614 Ki > 2000 nM T67363 C5PSA8 44305637 Ki > 10000 nM T67363 C4RMV1 44305685 Ki > 10000 nM T67363 C16EAZ 44305736 Ki > 2000 nM T67363 CD3R1S 44305804 Ki = 200 nM T67363 CQO62G 44306081 Ki = 1100 nM T67363 CS67MW 44320027 IC50 = 1.4 nM T67363 C91SAN 44320056 IC50 = 6.8 nM T67363 CC4UG8 44320077 IC50 = 3.6 nM T67363 CAVD13 44320155 IC50 = 0.3 nM T67363 C95KAZ 44320173 IC50 = 1.4 nM T67363 CSV1C2 44320174 IC50 = 0.38 nM T67363 C7GXI5 44320211 IC50 = 0.063 nM T67363 CWS24X 44320274 IC50 = 0.59 nM T67363 C1W8ID 44320282 IC50 = 0.22 nM T67363 C6F7OI 44320305 IC50 = 0.15 nM T67363 CN08CV 44320306 IC50 = 0.056 nM T67363 CVX0F7 44320364 IC50 = 0.16 nM T67363 CKY2F1 44329896 Ki > 1000 nM T67363 CKXQ61 44329897 Ki > 1000 nM T67363 C79CIF 44329957 IC50 = 8.8 nM T67363 C91OLV 44329959 IC50 = 2.9 nM T67363 CUQ2M9 44330009 IC50 = 12 nM T67363 CUK74V 44330015 Ki = 0.1 nM T67363 C38PGY 44330039 Ki = 10 nM T67363 CF9SY3 44330086 Ki = 7.3 nM T67363 CL7X1Y 44330191 Ki = 2.4 nM T67363 CAT6Y2 44330200 Ki = 154 nM T67363 C84HUN 44330327 Ki = 2.9 nM T67363 CS5R8Y 44330343 Ki = 52.7 nM T67363 CSIG14 44333548 IC50 = 45 nM T67363 C2E3VH 44333550 IC50 = 2.5 nM T67363 C23DVQ 44333621 IC50 = 560 nM T67363 C4X3KB 44333751 IC50 = 0.58 nM T67363 CY84IA 44333752 IC50 = 1400 nM T67363 CLE04Q 44333753 IC50 = 5.5 nM T67363 C2Y1DN 44337387 Ki = 3 nM T67363 C7UNY0 44337391 Ki = 30 nM T67363 CXE0S1 44337395 Ki = 9 nM T67363 CPKS69 44337398 Ki = 750 nM T67363 C49AYH 44337411 Ki = 5.5 nM T67363 C3CH4K 44337416 Ki = 4 nM T67363 C9W6XI 44337484 Ki = 2.5 nM T67363 C59DSH 44337494 Ki = 28 nM T67363 CFX1T4 44337503 Ki = 3 nM T67363 COA3Q4 44337517 Ki = 20 nM T67363 C75CFE 44337554 Ki = 2.5 nM T67363 CY7B9I 44337558 Ki = 90 nM T67363 CGF12D 44337568 Ki = 50 nM T67363 CF98VE 44337590 Ki = 710 nM T67363 CSU14K 44337595 Ki = 4 nM T67363 CD0FP8 44337598 Ki = 19 nM T67363 C6GA9C 44337603 Ki = 19 nM T67363 CKCD52 44337614 Ki = 6 nM T67363 C7HM5E 44337619 Ki = 23 nM T67363 CGOZ02 44337626 Ki = 10 nM T67363 CJC8A9 44337648 Ki = 15 nM T67363 C9A1QD 44337653 Ki = 13 nM T67363 CP75DF 44337654 Ki = 15 nM T67363 CJQB24 44337666 Ki = 2.5 nM T67363 CZ0YE1 44337684 Ki = 4 nM T67363 CDLE79 44337733 Ki = 2900 nM T67363 CN0K7Q 44337734 Ki = 1100 nM T67363 CY5R8E 44337742 Ki = 480 nM T67363 CAQZ60 44337758 Ki = 5 nM T67363 C6AZ8M 44337770 Ki = 9 nM T67363 CA47BJ 44337773 Ki = 70 nM T67363 CV37XE 44337781 Ki = 11 nM T67363 C8R0IV 44337782 Ki = 1300 nM T67363 CKN15C 44337788 Ki = 2 nM T67363 CYI89D 44337808 Ki = 14 nM T67363 CH6U5P 44337809 Ki = 8.5 nM T67363 CAHO14 44337810 Ki = 2.5 nM T67363 C82QTV 44337813 Ki = 180 nM T67363 CX0Q3S 44337817 Ki = 6.5 nM T67363 CB7H1S 44337824 Ki = 13 nM T67363 CKLC52 44337827 Ki = 27 nM T67363 C8KDE7 44337828 Ki = 10 nM T67363 C2A8MH 44337853 Ki = 15 nM T67363 CY2K0F 44337919 Ki = 1.9 nM T67363 C4LEU0 44340569 IC50 = 68 nM T67363 CTRQ17 44341096 IC50 = 597000 nM T67363 C6W4MS 44342344 IC50 = 5.8 nM T67363 CM20KE 44342349 IC50 = 1.1 nM T67363 C6CFS9 44342350 IC50 = 230 nM T67363 CWJ50A 44342406 IC50 = 29 nM T67363 CK9S6J 44342476 IC50 = 3.7 nM T67363 CIW85X 44342619 IC50 = 2.2 nM T67363 CSK3O5 44342624 IC50 = 4 nM T67363 CX46NY 44343237 IC50 = 1000 nM T67363 CDI59B 44344027 IC50 = 57.4 nM T67363 CIVR98 44344134 IC50 = 84 nM T67363 C7HLM3 44344166 IC50 = 0.35 nM T67363 C3R6QE 44344237 IC50 = 0.29 nM T67363 CF61PZ 44344250 IC50 = 0.49 nM T67363 CTOM36 44344252 IC50 = 0.74 nM T67363 CELV48 44350342 IC50 = 49 nM T67363 CP4R1A 44350344 IC50 = 180 nM T67363 CDE56C 44350392 IC50 = 41 nM T67363 CEP6G1 44350415 IC50 = 87 nM T67363 C7J9NH 44350447 IC50 = 57 nM T67363 CH6UX8 44350448 IC50 = 130 nM T67363 C4C2PF 44350449 IC50 = 32 nM T67363 CP4TD3 44350450 IC50 = 34 nM T67363 C9FUW5 44352004 IC50 = 130 nM T67363 CZB1K3 44358085 IC50 = 0.6 nM T67363 CBHY62 44358770 IC50 = 1000 nM T67363 CB6PL8 44358778 IC50 = 500 nM T67363 CCX8Y2 44358809 IC50 = 10000 nM T67363 CQ25DK 44358812 IC50 = 5000 nM T67363 C2BQO4 44358831 IC50 = 10000 nM T67363 C0L7WE 44358833 IC50 = 84 nM T67363 CTQP52 44358841 IC50 = 220 nM T67363 C15YTW 44358897 IC50 = 380 nM T67363 C3JPK8 44359000 IC50 = 10000 nM T67363 CVK7C1 44359080 IC50 = 12.9 nM T67363 C3XY7F 44359081 IC50 = 14.9 nM T67363 C8LO0N 44359086 IC50 = 1000 nM T67363 CZ7YE0 44359087 IC50 = 1000 nM T67363 CIPX97 44359766 IC50 = 140 nM T67363 CNLV75 44359767 IC50 = 320 nM T67363 CNZQ89 44366409 IC50 = 0.11 nM T67363 C1J2CW 44366410 IC50 = 3.3 nM T67363 CB0TF6 44368570 IC50 = 0.04 nM T67363 C47OWF 44368757 IC50 = 0.35 nM T67363 CV2K3S 44369353 IC50 = 55 nM T67363 CW0O4B 44369428 IC50 = 51 nM T67363 C32OCG 44369435 IC50 = 250 nM T67363 CK9WF1 44369491 IC50 = 25 nM T67363 CO83JW 44369641 IC50 = 7.3 nM T67363 CKRS68 44369648 IC50 > 1000 nM T67363 CAS01N 44372658 IC50 = 4200 nM T67363 CGIP26 44372909 IC50 = 300 nM T67363 CYD6H2 44372941 IC50 = 5800 nM T67363 C4NU0I 44372954 IC50 = 200 nM T67363 C6B5FO 44372955 IC50 = 800 nM T67363 CFO34W 44372962 IC50 = 5000 nM T67363 C0FAJ9 44372963 IC50 = 5900 nM T67363 C83JEF 44372972 IC50 = 9600 nM T67363 COYQ79 44372977 IC50 = 4500 nM T67363 C9C8LB 44373013 IC50 = 10600 nM T67363 CRV01L 44373014 IC50 = 11200 nM T67363 C1H3KN 44373023 IC50 > 30000 nM T67363 CHS2V0 44373024 IC50 = 4200 nM T67363 CBY0V9 44373073 IC50 = 15200 nM T67363 CNDV21 44373074 IC50 = 14300 nM T67363 CH1KV2 44373098 IC50 = 29600 nM T67363 CX9G4K 44373132 IC50 > 30000 nM T67363 C8WQ3F 44373152 IC50 = 1800 nM T67363 C9GH8E 44373158 IC50 = 5800 nM T67363 CFGE74 44373159 IC50 > 30000 nM T67363 CNX95Q 44373169 IC50 = 9200 nM T67363 CKR0X7 44373170 IC50 = 200 nM T67363 C6X9UK 44373176 IC50 = 2900 nM T67363 CAIJ06 44373182 IC50 = 120 nM T67363 C09MLI 44373256 IC50 = 4000 nM T67363 CB7UV8 44373257 IC50 = 1500 nM T67363 C89GTD 44373300 IC50 = 10000 nM T67363 CU12HA 44373303 IC50 = 2600 nM T67363 C68DAQ 44373341 IC50 = 4000 nM T67363 CQE4R3 44373603 IC50 = 2900 nM T67363 C9LWK0 44373604 IC50 = 25000 nM T67363 C4V3KU 44373605 IC50 = 3800 nM T67363 CWDC18 44383692 IC50 = 2600 nM T67363 CAY53C 44383697 IC50 = 96 nM T67363 CB2KW6 44383745 IC50 = 900 nM T67363 C3Q0GH 44383752 IC50 = 180 nM T67363 CBH12Q 44383755 IC50 = 140 nM T67363 CP1QH2 44383802 IC50 = 23 nM T67363 CY70ZS 44383803 IC50 = 12 nM T67363 CRJ1M9 44383805 IC50 = 480 nM T67363 CCR0M8 44383848 IC50 = 87 nM T67363 C1E0CL 44384154 IC50 = 14 nM T67363 C28CSF 44384225 IC50 = 16 nM T67363 CG0I7U 44384233 IC50 = 4 nM T67363 C3VKC9 44384418 IC50 = 36 nM T67363 CWY40J 44384448 IC50 = 300 nM T67363 CWX1O8 44384452 IC50 = 470 nM T67363 CR51GC 44384509 IC50 = 710 nM T67363 C2PXN3 44384519 IC50 = 310 nM T67363 C1SKZ8 44384644 IC50 = 8 nM T67363 CBV4X3 44384707 IC50 = 24 nM T67363 C1U0OM 44384812 IC50 = 23 nM T67363 CD95EQ 44384863 IC50 = 110 nM T67363 C7WK9L 44384982 IC50 = 100 nM T67363 C3ZCI0 44385023 IC50 = 66 nM T67363 CZIJ16 44385402 IC50 = 72 nM T67363 C54ZFB 44386844 Ki = 60 nM T67363 C0I4EG 44387184 IC50 = 1.9 nM T67363 CU98AB 44393368 IC50 > 20000 nM T67363 CVYB52 44393453 IC50 = 100 nM T67363 CBM2H6 44393479 IC50 = 9 nM T67363 CLR2T1 44393484 IC50 = 10.5 nM T67363 CH68MD 44393496 IC50 > 20000 nM T67363 C8YE7I 44393515 IC50 > 20 nM T67363 CAD12L 44393517 IC50 = 6.1 nM T67363 CV50SI 44393535 IC50 = 7.2 nM T67363 C5FVM2 44393536 IC50 > 20000 nM T67363 CM15VE 44393587 IC50 = 310 nM T67363 CEZB32 44393807 IC50 = 2.3 nM T67363 CD17AF 44393819 IC50 = 0.8 nM T67363 C4UF6A 44393849 IC50 = 0.4 nM T67363 CI5BK2 44393875 IC50 = 73.8 nM T67363 CG0VY1 44394008 IC50 = 0.8 nM T67363 CD6B3E 44394057 IC50 = 0.1 nM T67363 CS2I9D 44394317 IC50 = 3.4 nM T67363 CL9GN5 44394834 IC50 = 2.8 nM T67363 CIS4X5 44394933 IC50 = 21.7 nM T67363 CA30XW 44394981 IC50 = 25.3 nM T67363 C4X2PI 44395065 IC50 = 2.6 nM T67363 C0IN2J 44395933 IC50 = 0.8 nM T67363 CL1AJ8 44395975 IC50 = 2.6 nM T67363 CK4YH8 44396023 IC50 = 0.5 nM T67363 C3DN8C 44396062 IC50 = 1.2 nM T67363 C60IFP 44396497 IC50 = 7.2 nM T67363 CU1FH2 44399412 IC50 = 130 nM T67363 C5M8DS 44399508 IC50 = 8 nM T67363 CH3M9D 44399616 IC50 = 0.3 nM T67363 C8GE7Y 44399670 IC50 > 20000 nM T67363 C95SQZ 44399673 IC50 = 0.26 nM T67363 CDKW31 44399720 IC50 > 20000 nM T67363 CNJ6U7 44399721 IC50 = 0.25 nM T67363 CE18LD 44407524 IC50 = 1.28 nM T67363 CZ4O2D 44407529 IC50 = 0.62 nM T67363 CV36MS 44407555 IC50 = 2 nM T67363 C9XIY5 44407556 IC50 = 1.1 nM T67363 C1E7HF 44407560 IC50 = 0.74 nM T67363 CW8MQ7 44407577 IC50 = 2.4 nM T67363 C03KFP 44407668 IC50 = 1.2 nM T67363 C7CP1X 44407779 IC50 = 4 nM T67363 CB5R4A 44408398 IC50 > 1000 nM T67363 C43TRL 44408407 IC50 > 1000 nM T67363 C5LF3K 44412296 IC50 = 21 nM T67363 CZ7Q2H 44423872 IC50 = 0.5 nM T67363 CKQ84P 44423882 IC50 = 0.5 nM T67363 C4Z5QK 44423888 IC50 = 472 nM T67363 C8CM2P 44423899 IC50 = 12 nM T67363 C4R7IN 44429070 IC50 = 3 nM T67363 C8PJH9 44429072 IC50 = 0.9 nM T67363 CU4ME6 44429074 IC50 = 4 nM T67363 C2XN7B 44429081 IC50 = 0.7 nM T67363 CZ05RQ 44429084 IC50 = 1 nM T67363 C2EPI3 44429086 IC50 = 1 nM T67363 CHMJ47 44429089 IC50 = 1 nM T67363 CAK98T 44429091 IC50 = 10 nM T67363 C7J9AT 44429095 IC50 = 5 nM T67363 C0IUL1 44429100 IC50 = 5 nM T67363 C2IEY6 44429103 IC50 = 0.6 nM T67363 CC6FH0 44429107 IC50 = 1 nM T67363 CY1NM2 44429112 IC50 = 1 nM T67363 CE6WM2 44429118 IC50 = 5 nM T67363 CVW52C 44429121 IC50 = 0.7 nM T67363 C78CKB 44429123 IC50 = 0.4 nM T67363 C0Y9RK 44429125 IC50 = 3 nM T67363 C7CNA1 44429126 IC50 = 10 nM T67363 C7IO1Q 44429128 IC50 = 8 nM T67363 CC2Q8N 44429141 IC50 = 2.7 nM T67363 CW7HB6 44429142 IC50 = 8 nM T67363 C07LGP 44429143 IC50 = 1 nM T67363 CEW73I 44429144 IC50 = 2 nM T67363 CAX24B 44429145 IC50 = 3 nM T67363 CYV86W 44429146 IC50 = 33 nM T67363 C1PE8W 44429147 IC50 = 21 nM T67363 C8PTR0 44429148 IC50 = 20 nM T67363 CR58CB 44429149 IC50 = 4 nM T67363 C87WFU 44429150 IC50 = 10 nM T67363 CG6H7J 44429151 IC50 = 2 nM T67363 C8TNX7 44429152 IC50 = 3 nM T67363 CD1IN9 44429153 IC50 = 7 nM T67363 C7MTE0 44429154 IC50 = 9 nM T67363 CAS34H 44429155 IC50 = 7 nM T67363 C89OWZ 44429156 IC50 = 3 nM T67363 C4K0NT 44429157 IC50 = 1 nM T67363 C0C9KL 44429158 IC50 = 1 nM T67363 CVSI23 44429159 IC50 = 0.3 nM T67363 CEHF56 44429160 IC50 = 3 nM T67363 C8E3SH 44429161 IC50 = 18 nM T67363 CT47WG 44429162 IC50 = 54 nM T67363 CA01YX 44429163 IC50 = 10 nM T67363 CTM39A 44429164 IC50 = 5 nM T67363 CGQU48 44429165 IC50 = 56 nM T67363 CF5U9Z 44429166 IC50 = 5 nM T67363 COU58G 44429167 IC50 = 11 nM T67363 CN8GI9 44429168 IC50 = 13 nM T67363 C6G7RF 44436701 IC50 > 1000000 nM T67363 CZ1L9O 44436703 IC50 > 1000000 nM T67363 C7CAJ3 44436705 IC50 = 240 nM T67363 CR6XE2 44436707 IC50 = 21000 nM T67363 CYOC34 44436708 IC50 > 1000000 nM T67363 CSF3V2 44436709 IC50 = 120000 nM T67363 C67VHW 44436710 IC50 > 1000000 nM T67363 CBW09N 44436711 IC50 > 1000000 nM T67363 CRNQ31 44436712 IC50 > 1000000 nM T67363 C1YMJ2 44436713 IC50 = 600 nM T67363 CF4UR2 44436714 IC50 = 45000 nM T67363 C52DMG 44436715 IC50 > 1000000 nM T67363 CLU84X 44436716 IC50 = 15100 nM T67363 CRO80K 44436717 IC50 = 71 nM T67363 CQL95B 44439573 IC50 = 150 nM T67363 CVHD90 44439574 IC50 = 100000 nM T67363 CA6T8P 44439577 IC50 = 230000 nM T67363 C4A7UK 44439578 IC50 > 100000 nM T67363 CJ26IQ 44439579 IC50 = 2600 nM T67363 CJ82ND 44439580 IC50 = 35 nM T67363 CAJS34 44439581 IC50 = 20000 nM T67363 C4SD5P 44439582 IC50 = 1200 nM T67363 C3AH5M 44444138 Ki = 700 nM T67363 C2U4DR 44444139 Ki = 400 nM T67363 CA46OD 44444140 Ki > 2000 nM T67363 CHYP37 44444141 Ki = 650 nM T67363 CB0X8K 44444142 Ki = 33 nM T67363 CCTS86 44444143 Ki = 1.3 nM T67363 CWZX26 44444144 Ki = 11 nM T67363 C39TCU 44444145 Ki = 25 nM T67363 CE6WX7 44444146 Ki = 10 nM T67363 C0X8SG 44444147 Ki = 0.1 nM T67363 CSG83Z 44454980 IC50 = 122 nM T67363 CWIY29 44454981 IC50 = 10000 nM T67363 CJI3K2 44455003 IC50 = 500 nM T67363 CMA70X 44455005 IC50 = 50 nM T67363 C7P0QS 44455006 IC50 = 1000 nM T67363 C1RF6O 44455037 IC50 = 10 nM T67363 CM60TK 44455039 IC50 = 13 nM T67363 CN0Z4F 44455040 IC50 = 37 nM T67363 C87QUH 44455076 IC50 = 4.2 nM T67363 CB8AQ5 44455077 IC50 = 5000 nM T67363 CP13IF 44455109 IC50 = 27 nM T67363 CZO28A 44455111 IC50 = 7.4 nM T67363 CSJU52 44455112 IC50 = 50 nM T67363 CSN1G9 44455149 IC50 = 4.4 nM T67363 C94VDZ 44455151 IC50 = 1.5 nM T67363 CMVN47 44455456 IC50 = 10000 nM T67363 CMR2F1 44459058 IC50 > 100000 nM T67363 C13NVH 44459345 IC50 > 100000 nM T67363 CDKG38 44459361 IC50 > 100000 nM T67363 C9G5ZA 44459507 IC50 > 100000 nM T67363 C70KPC 44459508 IC50 > 100000 nM T67363 CX4JZ1 44459666 IC50 > 100000 nM T67363 C6O8ZD 44459743 IC50 > 100000 nM T67363 CAXJ53 44459773 IC50 > 100000 nM T67363 CU95CL 44459843 IC50 > 100000 nM T67363 CFJC10 44459851 IC50 > 100000 nM T67363 CGJ3Y7 44459852 IC50 > 100000 nM T67363 C56CVI 44459873 IC50 > 100000 nM T67363 C9CAP7 44459874 IC50 > 100000 nM T67363 CO3MN2 44460983 IC50 = 13.1 nM T67363 CJ54YG 44461075 IC50 = 3.3 nM T67363 CFT1K5 44461322 IC50 = 5.8 nM T67363 C4FSG2 44461379 IC50 = 5.9 nM T67363 CVDR72 44461391 IC50 = 0.67 nM T67363 C3BM9P 44461393 IC50 = 22.8 nM T67363 C0PFJ9 44461394 IC50 = 1.5 nM T67363 CY4L8W 44549109 IC50 = 0.5 nM T67363 C4FW5Y 44549223 IC50 = 0.8 nM T67363 C7IXB3 44550126 IC50 = 3.9 nM T67363 CW9N7S 44550127 IC50 = 0.8 nM T67363 CK4UM8 44550445 IC50 = 428 nM T67363 C3QU6T 44550446 IC50 = 1.2 nM T67363 CS0Z3D 44550447 IC50 = 1.4 nM T67363 CH9M4W 44550573 IC50 = 0.6 nM T67363 C5V7GK 44550574 IC50 = 1.7 nM T67363 CB7R0U 44550575 IC50 = 7.6 nM T67363 CN3T7E 44550576 IC50 = 1.7 nM T67363 CO8EM6 44550577 IC50 = 0.1 nM T67363 C4XF2A 44550689 IC50 = 1.1 nM T67363 C4T6XP 44550690 IC50 = 0.7 nM T67363 CUWQ62 44550691 IC50 = 0.6 nM T67363 C69RIT 44550947 IC50 = 0.9 nM T67363 CX1C4T 44552445 IC50 = 6.1 nM T67363 CJM54V 44580934 IC50 = 11.19 nM T67363 C27WPD 44580937 IC50 = 78.96 nM T67363 CTO29I 44591126 IC50 = 230 nM T67363 C4U9VF 44591153 IC50 = 180 nM T67363 CER2H0 44591154 IC50 = 39 nM T67363 C7TX9N 44591155 IC50 = 370 nM T67363 CCFW92 44605870 IC50 = 2000 nM T67363 C63TSK 44606191 IC50 = 3.9 nM T67363 CT0PO4 44606192 IC50 = 3.2 nM T67363 CM9VI1 44626482 IC50 = 920 nM T67363 CBO95I 44626483 IC50 > 100000 nM T67363 CS36GK 44627949 IC50 = 11000 nM T67363 CX6LM3 44628051 IC50 = 180 nM T67363 CVTO84 44628052 IC50 = 2300 nM T67363 CJQ37N 44628053 IC50 > 100000 nM T67363 CV4P3J 44628054 IC50 > 100000 nM T67363 CTU9W0 44628055 IC50 > 100000 nM T67363 CFMW09 45104120 Ki = 19.1 nM T67363 CHPW08 45104215 Ki = 14.8 nM T67363 C9RHC0 45483715 IC50 = 138 nM T67363 C4E8LZ 45483796 IC50 = 0.3 nM T67363 CU58DV 45483797 IC50 = 0.7 nM T67363 C18VUC 45483798 IC50 = 0.3 nM T67363 C5PZ8G 46201042 IC50 = 6.01 nM T67363 C89ZFA 46224777 IC50 = 89 nM T67363 C5X1NZ 46224858 IC50 = 614 nM T67363 CDG6B1 46224859 IC50 = 16600 nM T67363 CKM2X1 46224860 IC50 = 4.3 nM T67363 CL39GY 46224861 IC50 = 13.4 nM T67363 C56PVC 46226894 IC50 = 16000 nM T67363 CVXH79 46226896 IC50 = 319 nM T67363 CBKZ57 46226897 IC50 = 100 nM T67363 C30JXH 46226899 IC50 = 472 nM T67363 C2WHK1 46226900 IC50 = 1734 nM T67363 C5H9YT 46226901 IC50 = 2925 nM T67363 CV8W7P 46226902 IC50 = 1600 nM T67363 C83EWD 46226903 IC50 = 2423 nM T67363 CRVU54 46226904 IC50 = 890 nM T67363 CE85AX 46226905 IC50 = 261 nM T67363 C81VUL 46229417 IC50 = 0.59 nM T67363 CNP0O2 46229418 IC50 = 37.6 nM T67363 CPB51X 46229419 IC50 = 7.27 nM T67363 CC6HP8 46229421 IC50 = 3100 nM T67363 C1CR9Y 46229422 IC50 = 11.66 nM T67363 CR53AM 46229424 IC50 = 3.8 nM T67363 C0Y1TB 46232105 IC50 = 0.48 nM T67363 CJ06HG 46232379 Ki = 2.9 nM T67363 CSI0V2 46232380 Ki = 2 nM T67363 C81NZJ 49782807 IC50 > 10000 nM T67363 C17UYM 49782809 IC50 > 10000 nM T67363 CNT47C 49782811 IC50 > 10000 nM T67363 CK52QA 49782813 IC50 > 10000 nM T67363 CCX41K 49783020 IC50 = 1.35 nM T67363 CEW9Q0 50899825 IC50 = 0.09 nM T67363 CP7U9T 50907449 IC50 > 1000 nM T67363 C59LHA 52941929 IC50 > 10000 nM T67363 C04OYX 52942589 IC50 > 10000 nM T67363 C69YHV 52943199 IC50 > 10000 nM T67363 C8AS0O 52943382 IC50 = 4960 nM T67363 C3OTG8 52944258 IC50 = 0.16 nM T67363 CE9DO8 52944259 IC50 = 0.11 nM T67363 C2ADU0 52944260 IC50 = 0.32 nM T67363 CEF0A3 52945622 IC50 > 10000 nM T67363 CGLR93 52946695 IC50 = 0.16 nM T67363 CVDT37 52946696 IC50 = 0.16 nM T67363 C7MW0D 52948102 IC50 = 1350 nM T67363 C5T8DB 52948257 IC50 > 10000 nM T67363 C5K2ME 52948941 IC50 > 10000 nM T67363 CF10XI 52949257 IC50 > 10000 nM T67363 CV9B3M 52950165 IC50 = 3470 nM T67363 CM2VX7 53317165 EC50 = 2.5 nM T67363 C6XNM0 53380822 IC50 > 100000 nM T67363 C1KFQ0 53380823 IC50 > 100000 nM T67363 C7JWD0 53380936 IC50 > 100000 nM T67363 C97KGD 53380937 IC50 > 100000 nM T67363 CKV6Q2 53380938 IC50 > 100000 nM T67363 C47WIH 53380939 IC50 > 100000 nM T67363 CY3RO0 53380940 IC50 > 100000 nM T67363 C3R8PW 53380941 IC50 > 100000 nM T67363 C2G6VQ 54580191 IC50 = 0.3 nM T67363 C1D8YQ 54581193 IC50 = 0.44 nM T67363 C6RSP2 54582337 IC50 = 720 nM T67363 C5Y8PF 54582338 IC50 > 10000 nM T67363 C0YTW6 54583189 IC50 = 0.25 nM T67363 CYRU74 54583322 IC50 = 4600 nM T67363 C7WEU3 54583323 IC50 > 10000 nM T67363 C75WYX 54584281 IC50 > 10000 nM T67363 CY08RT 54586079 IC50 = 0.17 nM T67363 C6OI5V 56660094 IC50 > 100000 nM T67363 CKFI81 56660095 IC50 > 100000 nM T67363 CT7U8L 56683905 IC50 > 100000 nM T67363 C3CDB4 56683906 IC50 > 100000 nM T67363 CK7ZI0 56838719 IC50 = 8800 nM T67363 CB57DW 57391171 IC50 > 100000 nM T67363 CWJ4I7 57391565 IC50 > 100000 nM T67363 C7APO2 57392934 IC50 > 100000 nM T67363 CZ2A0S 57392935 IC50 > 100000 nM T67363 CX16KB 57393324 IC50 > 100000 nM T67363 C6EWL9 57394677 IC50 > 100000 nM T67363 C8T2ZJ 57395044 IC50 > 100000 nM T67363 C9F4OL 57398232 IC50 > 100000 nM T67363 C5OAB7 57398233 IC50 > 100000 nM T67363 CY39KP 57398234 IC50 > 100000 nM T67363 CODX48 57399879 IC50 > 100000 nM T67363 C93VSX 57399880 IC50 > 100000 nM T67363 C5WOZ3 57399881 IC50 > 100000 nM T67363 C9ZL5X 57400230 IC50 > 100000 nM T67363 CPZR79 57400272 IC50 > 100000 nM T67363 CS2ZY1 57401658 IC50 > 100000 nM T67363 CG90KP 57403382 IC50 > 100000 nM T67363 C3CKA6 57403383 IC50 > 100000 nM T67363 C4OB6Z 57403384 IC50 > 100000 nM T67363 CKI4S8 57403776 IC50 > 100000 nM T67363 C94QEJ 57521432 IC50 = 7.6 nM T67363 CB86RW 57521433 IC50 = 0.2 nM T67363 C1RDQ5 57521434 IC50 = 2.1 nM T67363 CKHE62 57521435 IC50 = 0.2 nM T67363 CT7FL5 57523172 IC50 = 4.5 nM T67363 CR71ZG 59665343 IC50 = 23 nM T67363 C60EVZ 59665407 IC50 = 49 nM T67363 C4UH8X 59665418 IC50 = 1200 nM T67363 CSRE10 59665495 IC50 = 6700 nM T67363 C5HP9O 60154467 IC50 = 48 nM T67363 C1C0UT 68898764 IC50 = 8800 nM T67363 CN93KB 68898863 IC50 = 520 nM T67363 C9LB1Y 68900219 IC50 = 620 nM T67363 C74UPO 68900657 IC50 = 510 nM T67363 CF4BZ9 68901306 IC50 = 370 nM T67363 CI0AL7 69244056 IC50 = 340 nM T67363 CU65XM 69693295 IC50 = 1.995 nM T67363 C31IUF 69863577 IC50 > 10000 nM T67363 CQ4G2O 70683715 IC50 = 350 nM T67363 CPAQ48 70684198 Ki > 10000 nM T67363 CP8KD5 70686837 Ki = 0.663 nM T67363 CVCJ03 70687988 IC50 = 0.3 nM T67363 CX73MA 70689988 IC50 = 8300 nM T67363 C8NZ7A 70694228 IC50 = 17 nM T67363 C5G9BX 71449526 IC50 = 4.83 nM T67363 C1GAT7 71451321 IC50 = 1.3 nM T67363 CQ0U6Z 71451322 IC50 = 4.97 nM T67363 C4VP1N 71454873 IC50 = 800 nM T67363 CH4R2Z 71454874 IC50 = 2.3 nM T67363 C2TCV3 71454875 IC50 = 2.28 nM T67363 COJ71C 71454876 IC50 = 6.3 nM T67363 CZB06S 71456647 IC50 = 108.9 nM T67363 C23GSR 71459889 IC50 = 2800 nM T67363 C5Q3PB 71461030 IC50 = 4.1 nM T67363 C9DS7U 71461032 IC50 = 26.4 nM T67363 C8EM7Y 71550913 IC50 = 0.86 nM T67363 CY1MD5 71574157 IC50 > 10000 nM T67363 C02ZBI 71574158 IC50 = 675 nM T67363 C16JKI 71574159 IC50 > 10000 nM T67363 CU95LC 71574160 IC50 = 516 nM T67363 COJ8Y4 71574161 IC50 > 10000 nM T67363 C5SG9H 71574261 IC50 = 576 nM T67363 C3C9QK 71574262 IC50 = 3871 nM T67363 CTZU49 71574263 IC50 > 10000 nM T67363 C4HB7F 71574264 IC50 > 10000 nM T67363 C3S9QJ 71574355 IC50 > 10000 nM T67363 C8V4UB 71574356 IC50 > 10000 nM T67363 CX0SQ1 71574452 IC50 > 10000 nM T67363 C9J7NH 71652207 IC50 > 200000 nM T67363 CLH52G 71654374 IC50 > 200000 nM T67363 C8GDV7 71654376 IC50 > 200000 nM T67363 CY29LR 71654530 IC50 > 200000 nM T67363 C3K6PT 71654532 IC50 > 200000 nM T67363 C3X7FP 71654534 IC50 > 200000 nM T67363 CCGP56 71654535 IC50 > 200000 nM T67363 CZG3Y9 71654536 IC50 > 200000 nM T67363 C1QE0K 71716365 IC50 = 13.6 nM T67363 CFYM81 71720633 IC50 > 10000 nM T67363 CA9K6E 72204688 IC50 > 100000 nM T67363 CLC7R0 72204689 IC50 = 1490 nM T67363 CCW43J 72204873 IC50 = 830 nM T67363 CQ6TF8 72204875 IC50 = 120 nM T67363 CC49AN 72204878 IC50 > 100000 nM T67363 C0N3SX 72205060 IC50 = 270 nM T67363 C8B7QE 72949858 IC50 = 0.8 nM T67363 C0BJ1F 73345752 IC50 = 2 nM T67363 C4P3JC 73346588 IC50 = 10.62 nM T67363 C9UD8K 73346937 Ki = 10 nM T67363 C8X0BY 73347135 IC50 = 880 nM T67363 CP47JC 73348619 IC50 = 2.9 nM T67363 CF1UL2 73348680 IC50 = 24 nM T67363 C5BQ6R 73349139 IC50 = 71 nM T67363 C6WTA2 73350123 IC50 = 40 nM T67363 C0PU3D 73351771 IC50 = 4 nM T67363 CM94NF 73353043 IC50 = 98100 nM T67363 C2SYT7 73353316 IC50 = 0.6 nM T67363 CN1P5F 73354828 IC50 = 6 nM T67363 CC19KU 73356070 Ki = 10 nM T67363 CO3WF4 73356277 IC50 = 840 nM T67363 CXM8L3 75002097 IC50 = 100 nM T67363 CD46SJ 76321533 IC50 > 100000 nM T67363 CNF56Z 76332375 IC50 > 100000 nM T67363 C30NBD 86272865 IC50 = 1000 nM T67363 CW8UV5 86272868 Ki = 39.81 nM T67363 CI07FE 90645591 IC50 = 21000 nM T67363 C8N6OE 90654504 IC50 = 0.65 nM T67363 C8TWH9 90654505 IC50 = 638 nM T67363 CDVB75 90654506 IC50 = 75.1 nM T67363 C5HG9N 90654507 IC50 = 1.6 nM T67363 CLCN89 117977916 IC50 = 160 nM T67363 CJO3B6 117978172 IC50 > 10000 nM T67363 C7ANO1 118709464 IC50 = 87 nM T67363 C2J3VA 118721315 IC50 = 316.23 nM T67363 C0BT3F 118721316 IC50 = 1995.26 nM T67363 C4TNZ0 118721317 IC50 = 50.12 nM T67363 C2N6WI 118721318 IC50 = 501.19 nM T67363 CMQ94S 118721319 IC50 = 79.43 nM T67363 C5CW9O 118721320 IC50 = 158.49 nM T67363 CYL2X3 118721321 IC50 = 39.81 nM T67363 CFQA95 118721322 IC50 = 100 nM T67363 CWDE71 118721323 IC50 = 125.89 nM T67363 CM9J4X 118721324 IC50 = 39.81 nM T67363 CY13BE 118721325 IC50 = 25.12 nM T67363 C8UNZ5 118721326 IC50 = 79.43 nM T67363 CG5B9F 118721327 IC50 = 251.19 nM T67363 CMXJ63 118721328 IC50 = 158.49 nM T67363 C2OJX9 118721329 IC50 = 125.89 nM T67363 C0YG4M 118721330 IC50 = 100 nM T67363 C8F4DG 118721331 IC50 = 199.53 nM T67363 C2ESU9 118721332 IC50 = 199.53 nM T67363 C2OYU9 118721333 IC50 = 100 nM T67363 CX0R3H 118721334 IC50 > 10000 nM T67363 CP8I3D 118721335 IC50 = 398.11 nM T67363 CGM28Y 118721336 IC50 = 3981.07 nM T67363 COM73D 118721337 IC50 = 50.12 nM T67363 CH25GR 118721338 IC50 = 125.89 nM T67363 CE7D1S 118721339 IC50 = 63.1 nM T67363 CZ95CL 118721340 IC50 = 125.89 nM T67363 C0AL1C 118721341 IC50 = 398.11 nM T67363 CAZ6U3 118721342 IC50 = 100 nM T67363 C65KQW 118721343 IC50 = 1584.89 nM T67363 COW6E1 118731284 IC50 = 50000 nM T67363 COE40F 118731285 IC50 = 100000 nM T67363 CG6WF1 118731286 IC50 > 100000 nM T67363 CHD10T 118753906 IC50 = 2 nM T67363 CE7PC8 118753907 IC50 = 7 nM T67363 CGJ9O5 118978102 IC50 = 630.96 nM T67363 CL2ER8 121242162 IC50 = 125.89 nM T67363 CPS9N3 121245322 IC50 = 1995.26 nM T67363 C8P7OW 121245346 IC50 = 3162.28 nM T67363 CJ83VH 121245350 IC50 = 10000 nM T67363 CFOM46 121246727 IC50 = 316.23 nM T67363 CL5Q9G 121246911 IC50 = 501.19 nM T67363 CAL43C 121246982 IC50 = 1258.93 nM T67363 C6XK2Y 121247103 IC50 = 50.12 nM T67363 CV7DK0 122181680 IC50 > 1000 nM T67363 CWY3V2 122181682 IC50 > 1000 nM T67363 CRG07Q 124155531 IC50 > 10000 nM T67363 C69XPN 124163720 IC50 > 10000 nM T67363 C4R3BT 124163838 IC50 = 2000 nM T67363 CS2QR4 124163840 IC50 = 4000 nM T67363 C93HFX 127025140 IC50 = 34 nM T67363 CEU4X3 127025441 IC50 = 2.4 nM T67363 CTX71B 127025442 IC50 = 20 nM T67363 C2FZ5Y 127037453 IC50 = 221 nM T67363 CR5X1T 130453989 IC50 = 158.49 nM T67363 CVT2U3 130454024 IC50 = 158.49 nM T67363 CT4BY6 130454058 IC50 = 158.49 nM T67363 CZK41V 130454091 IC50 = 251.19 nM T67363 C2OJ3C 130454093 IC50 = 199.53 nM T67363 CU73IM 131985420 IC50 = 199.53 nM T67363 CQEK82 131985476 IC50 = 1000 nM T67363 C20ZAT 131985489 IC50 = 251.19 nM T67363 C1IKD6 131985494 IC50 = 251.19 nM T67363 CI6W9O 131985523 IC50 = 794.33 nM T67363 C57BQS 132561360 IC50 = 6309.57 nM T67363 CP98GA 132601202 IC50 = 0.497 nM T67363 C21ACR 133633869 IC50 = 29 nM T67363 C9J6BA 135498601 IC50 > 1000 nM T67363 CB63XI 135509541 IC50 = 52 nM T67363 CJL87N 135949396 IC50 = 1 nM T67363 CSCN42 135983770 IC50 = 2 nM T67363 CR8K5L 135983772 IC50 = 7 nM T67363 CVD0O1 136132281 IC50 = 130 nM T67363 CXZ16C 137480037 IC50 = 1000 nM T67363 CIL96B 137632126 IC50 = 152000 nM T67363 C1CPO0 137632555 IC50 = 257000 nM T67363 C85WBP 137634338 IC50 = 3.8 nM T67363 CMOI37 137641477 IC50 = 171000 nM T67363 CYS13G 137648507 IC50 = 33000 nM T67363 C4IX7Z 137649002 IC50 = 1.24 nM T67363 CDO0Q6 137650356 IC50 = 7200 nM T67363 C6NVW5 137652892 IC50 = 5.1 nM T67363 CTL61H 137655644 IC50 = 1800 nM T67363 C4GO5B 137661340 IC50 = 48800 nM T67363 CV6JY5 139030528 IC50 = 6309.57 nM T67363 CAK31T 139593557 IC50 = 3.981 nM T67363 C0X8ER 145949722 IC50 = 0.91 nM T67363 C1LA9J 145949829 Ki = 103 nM T67363 C2MO7K 145951845 IC50 = 0.21 nM T67363 CG80FB 145951878 IC50 = 1.3 nM T67363 C1P0NL 145952828 IC50 = 1.4 nM T67363 CJA7N9 145953608 IC50 = 1.7 nM T67363 CI4H5X 145953880 Ki = 19.9 nM T67363 CZ4SK6 145954275 IC50 = 1.2 nM T67363 CTA08K 145956036 IC50 = 2.2 nM T67363 CY5I1O 145956101 IC50 = 1.6 nM T67363 C8RAG3 145956154 IC50 = 4 nM T67363 CYU26X 145956418 Ki = 26.5 nM T67363 CCB51L 145956802 IC50 = 1.2 nM T67363 CTS5R3 145959048 IC50 = 2.8 nM T67363 CQ4ET5 145959752 IC50 = 0.79 nM T67363 C4HD9N 145960086 Ki = 21.6 nM T67363 CS6RH1 145961486 IC50 <= 150 nM T67363 CO0W4J 145961652 IC50 = 4.5 nM T67363 CAST83 145961761 IC50 <= 150 nM T67363 C23HZY 145971531 IC50 = 0.91 nM T67363 CH9UP3 145982517 IC50 = 398.11 nM T67363 CX0P5N 145982847 IC50 = 199.53 nM T67363 CL13NC 145982905 IC50 = 158.49 nM T67363 C4N5TW 145983050 IC50 = 501.19 nM T67363 CJ70YV 145984499 IC50 = 158.49 nM T67363 C4R5NQ 145984560 IC50 = 1995.26 nM T67363 CM9FS1 145985439 IC50 = 3981.07 nM T67363 CRA6D0 145985939 IC50 = 50.12 nM T67363 C75GFR 154734316 IC50 = 352 nM T67363 C8ZUJ5 154734319 IC50 > 1000 nM T67363 CB2X7V 155511318 IC50 = 12.59 nM T67363 C1MSP9 155512998 IC50 = 25100 nM T67363 C7LI4B 155514586 IC50 = 50.12 nM T67363 CSMQ36 155514765 IC50 = 7.943 nM T67363 C17RZG 155515221 IC50 = 5.4 nM T67363 CHT1J6 155515540 IC50 = 632 nM T67363 CQ5C4M 155516533 IC50 = 43 nM T67363 CAOY19 155516610 IC50 = 3.162 nM T67363 CQNC74 155517321 IC50 = 239 nM T67363 CE1D6N 155518125 IC50 = 1.995 nM T67363 C35OHK 155518750 IC50 = 398.11 nM T67363 CTA5S4 155518784 IC50 = 5011.87 nM T67363 CRIA18 155519034 IC50 = 59.2 nM T67363 C3S2YZ 155519712 IC50 = 36.2 nM T67363 CZY8F6 155520344 IC50 = 250000 nM T67363 CMF13G 155520959 IC50 = 3.981 nM T67363 CL5K1Z 155521171 IC50 = 125.89 nM T67363 CL7OU0 155521485 IC50 = 1.995 nM T67363 C9OR7L 155522422 IC50 = 39.81 nM T67363 C90YTQ 155526362 IC50 = 2.512 nM T67363 C9HB1M 155526953 IC50 = 579 nM T67363 C1C8ZV 155527608 IC50 = 24500 nM T67363 C2GJ5V 155527654 IC50 = 11100 nM T67363 CQ1G0D 155528127 IC50 = 38.9 nM T67363 CZ68AU 155528189 IC50 = 3.162 nM T67363 C2GSD7 155528224 IC50 = 491 nM T67363 CPIL79 155528977 IC50 = 14.9 nM T67363 CR90VY 155529944 IC50 = 2130 nM T67363 C58JIQ 155530986 IC50 = 64.6 nM T67363 CJZU81 155532583 IC50 = 17.7 nM T67363 C6LAW0 155533172 IC50 = 1.259 nM T67363 C9T6SE 155533508 IC50 = 65 nM T67363 CJ7O2X 155534687 IC50 = 343 nM T67363 C3QT6L 155534872 IC50 = 158.49 nM T67363 CS03LO 155538904 IC50 = 0.7943 nM T67363 CE1W5B 155540544 IC50 = 12589.25 nM T67363 CYW32T 155541264 IC50 = 7.943 nM T67363 CB96AH 155545672 IC50 = 6.31 nM T67363 C6TCP5 155546837 IC50 > 1000 nM T67363 C89CHT 155548525 IC50 = 8900 nM T67363 CJZ35U 155549685 IC50 = 1.995 nM T67363 C6D2SM 155550380 IC50 = 537 nM T67363 CWF98D 155552156 IC50 > 1000 nM T67363 CW5AV4 155552698 IC50 = 5.012 nM T67363 CV4DG6 155554134 IC50 = 5.012 nM T67363 CJ6L8S 155561029 IC50 = 4200 nM T67363 CC64PJ 155561080 IC50 = 19 nM T67363 C80PGY 155563043 IC50 = 41.3 nM T67363 CKRE58 155563328 IC50 > 10000 nM T67363 CEF3T8 155563936 IC50 = 104 nM T67363 CR57YC 155565132 IC50 = 109600 nM T67363 C98UME 155566748 IC50 = 95.2 nM T67363 C5GQX9 155567527 IC50 = 3.162 nM T67363 C1HNT9 155567705 IC50 = 3981.07 nM T67363 CYZ02H 155568897 IC50 = 5011.87 nM T67363 CY8S2L 155569251 IC50 > 1000 nM T67363 C9NH4F 155569254 IC50 = 34 nM T67363 C7Z4RD 155569291 IC50 = 6309.57 nM T67363 C5FR9J 44385169 IC50 = 140 nM T67363 CUAI47 56665424 IC50 = 193 nM T67363 CZ9D2V 90645090 EC50 = 55 nM T67363 CWA6N4 90645092 EC50 = 11 nM T67363 CA8W7Q 90645094 EC50 = 10440 nM T67363 D00YBU 10699123 IC50 = 10.31 nM T67363 D01AXA 11764797 IC50 = 25 nM T67363 D01BZH 11613122 IC50 = 44.7 nM T67363 D01MGI 11583738 IC50 = 0.26 nM T67363 D03KLT 24822283 IC50 = 0.16 nM T67363 D03YLY 24822953 IC50 = 0.47 nM T67363 D04WVG 11540460 IC50 = 7.2 nM T67363 D05AGK 11743533 IC50 > 1000 nM T67363 D05EWB 10416726 IC50 = 36.3 nM T67363 D05GXK 24822444 IC50 = 0.91 nM T67363 D05VEC 11712622 IC50 = 7.7 nM T67363 D06JLN 11518823 IC50 = 5.6 nM T67363 D06LKH 123811 IC50 = 750 nM T67363 D07QJD 24822784 IC50 = 7.01 nM T67363 D07SFV 44123804 IC50 = 157 nM T67363 D07UOF 44408450 IC50 = 19.75 nM T67363 D07WDB 104802 IC50 > 10000 nM T67363 D08CFM 11505585 IC50 = 285.3 nM T67363 D09PLA 11533023 IC50 = 4.6 nM T67363 D0A0KS 9851104 IC50 = 0.00028 ug.mL-1 T67363 D0B4JU 15409414 IC50 = 100 nM T67363 D0F7SE 44123805 IC50 = 6.5 nM T67363 D0G8JI 44409460 IC50 = 28.7 nM T67363 D0H4EK 11643340 IC50 = 704.4 nM T67363 D0H4NK 4780 IC50 > 200000 nM T67363 D0I5BY 9831456 IC50 = 35.5 nM T67363 D0J6SP 24824620 IC50 = 0.18 nM T67363 D0LF7W 11569720 IC50 = 132.9 nM T67363 D0LV6B 130667 IC50 = 210 nM T67363 D0M0BN 11636164 IC50 = 7237.9 nM T67363 D0M6NQ 10372586 IC50 = 18.8 nM T67363 D0O6DN 11584047 IC50 = 35.6 nM T67363 D0O9FL 24823110 IC50 = 0.08 nM T67363 D0P4RB 44409497 IC50 = 730 nM T67363 D0R3CY 9952958 Ki = 4 nM T67363 D0R9AD 558969 IC50 = 33.5 nM T67363 D0R9GW 11540715 IC50 = 51.4 nM T67363 D0R9SJ 44439175 IC50 = 1.4 nM T67363 D0SA4A 1354 IC50 = 190600 nM T67363 D0T1II 44409643 IC50 = 63.9 nM T67363 D0U2NV 44408397 IC50 = 1017.8 nM T67363 D0UE7H 11670104 IC50 = 9.93 nM T67363 D0V0JC 9986643 IC50 = 237.1 nM T67363 D0W6CJ 11656381 IC50 = 712.7 nM T67363 D0X4EE 10415998 IC50 = 20 nM T67363 D0Z6WZ 24822282 IC50 = 0.03 nM T95446 D0W0VD 3885 IC50 = 11000 nM T95446 CLK6I5 14631798 IC50 = 6300 nM T95446 C5R4LE 14631799 IC50 = 22000 nM T95446 C6NYI9 22899233 IC50 = 30000 nM T95446 CMOV75 118727359 IC50 = 32000 nM T95446 CV68LZ 118727360 IC50 = 19000 nM T95446 CP79QH 137632568 IC50 = 25000 nM T95446 C4L2CA 137641351 IC50 = 17000 nM T95446 CQ4EM8 137643157 IC50 = 9000 nM T95446 CT21CH 137659467 IC50 = 19000 nM T95446 C7W4YA 137662216 IC50 = 35000 nM T38581 CUS16Z 44584846 Ki = 492 nM T38581 CP2J8X 44584953 Ki = 188 nM T38581 CBX8K0 44584960 Ki = 433 nM T38581 C10KCB 44584961 Ki = 806 nM T38581 C1S6KQ 44584962 Ki = 649 nM T38581 CJ73BT 45486346 Ki = 85 nM T38581 C9ETC4 45486354 Ki = 173 nM T38581 CVPG40 45486356 Ki = 6.3 nM T38581 CSQ2K4 45486357 Ki = 3.6 nM T38581 C0ET8W 137630787 Ki = 0.12 nM T38581 D05JJL 44584947 Ki = 232 nM T38581 D0Y9PH 45486355 Ki = 1.6 nM T20053 D0E3TC 44259 IC50 = 0.856 nM T20053 D03BNU 59604787 IC50 > 10000 nM T20053 D0T3ME 156422 IC50 > 30000 nM T20053 CACS26 11561968 Ki > 2000 nM T20053 CU0E8O 11690457 Ki > 10000 nM T20053 CLS29B 46872626 IC50 > 10000 nM T20053 C8NA4L 53384644 IC50 > 30000 nM T20053 CV63UL 67240318 IC50 > 10000 nM T20053 CPHG43 135567142 IC50 = 2 nM T20053 C2MD1Q 155513187 IC50 > 10000 nM T03500 D00HNB 25419 IC50 = 121000 nM T03500 D04AIT 5280445 IC50 = 980 nM T03500 D0K8KX 5280343 IC50 = 10230 nM T03500 D05VZE 119031 IC50 = 10000 nM T03500 D06IPZ 49800096 IC50 = 8300 nM T03500 D0G1LL 74221072 IC50 = 270 nM T03500 D0N6ZA 74221131 IC50 = 3400 nM T03500 D0UM5R 74221070 IC50 = 71 nM T03500 D0T9HG 132519 Ki = 0.52 nM T03500 CY78XM 4218 Ki = 0.61 nM T03500 CZ45IU 4219 IC50 = 8.2 nM T03500 CIP1T0 78598 IC50 = 2000000 nM T03500 C4D7TS 448002 Ki = 4.3 nM T03500 CVO6E9 2741314 IC50 = 1000000 nM T03500 C8SE4K 2763839 IC50 = 355000 nM T03500 CMNJ91 2801266 IC50 = 5000000 nM T03500 CME24U 3649035 IC50 = 13000 nM T03500 CBN96T 4358655 IC50 > 100000 nM T03500 CVLS16 5319161 IC50 = 1200 nM T03500 CJG2B7 6476333 IC50 = 8220 nM T03500 CL5DH0 6479915 IC50 = 2750 nM T03500 CP7BG0 6852146 IC50 = 14 nM T03500 C0FQW9 7063077 Ki = 672 nM T03500 C5DGI9 9851911 IC50 = 5 nM T03500 CI8Z0R 9866250 IC50 = 0.24 nM T03500 C75DAZ 9885136 IC50 = 3.5 nM T03500 CSIB97 9896504 IC50 > 30000 nM T03500 C03GVA 9932290 Ki = 360 nM T03500 C05HGV 9955795 IC50 = 2.6 nM T03500 CC4WG3 9957228 Ki > 300000 nM T03500 C09LSY 9979489 Ki > 6023 nM T03500 CUA65C 9982414 IC50 = 0.95 nM T03500 CO0TX7 9993891 Ki > 300000 nM T03500 CM4AL0 10001331 IC50 = 400 nM T03500 CR7T3J 10009978 Ki = 390 nM T03500 CM52RO 10030422 IC50 = 8.2 nM T03500 CJR59P 10031295 Ki > 6023 nM T03500 CLZ87W 10051236 Ki = 223 nM T03500 CP9HE6 10091931 IC50 = 400 nM T03500 C0G7IY 10114318 Ki = 240 nM T03500 C78JHL 10116107 Ki = 300 nM T03500 CYU19P 10127901 Ki > 4040 nM T03500 CH0UW2 10129190 Ki > 6020 nM T03500 C7KR3Y 10136680 Ki = 89.13 nM T03500 CNU93J 10136924 Ki = 280 nM T03500 C1CDF2 10136925 Ki = 346.74 nM T03500 CJ9EX4 10138303 Ki = 360 nM T03500 CFXC89 10139040 Ki > 5025 nM T03500 CO6PS3 10162900 Ki = 338.84 nM T03500 CR5H6E 10163627 IC50 = 250 nM T03500 CGB27E 10174981 Ki > 6020 nM T03500 CL47AR 10175070 Ki > 6020 nM T03500 C4ULO6 10175077 Ki > 6020 nM T03500 C84ZQD 10175219 Ki = 130 nM T03500 CIT0H4 10175323 Ki > 6020 nM T03500 C95IGP 10175331 Ki = 1020 nM T03500 CT7U0M 10175426 Ki > 6020 nM T03500 CCX3T6 10183064 Ki = 410 nM T03500 CK0P3F 10186536 IC50 = 540 nM T03500 C51RPY 10195069 Ki > 6020 nM T03500 CCHX74 10195307 Ki = 210 nM T03500 C94KHT 10195527 Ki > 6020 nM T03500 CDG35O 10196192 Ki = 390 nM T03500 CE1LI3 10204303 Ki = 480 nM T03500 CQFP69 10206106 Ki = 436.52 nM T03500 C4K1MJ 10208262 IC50 = 390 nM T03500 CG8FA4 10218128 Ki > 6020 nM T03500 C7Y2US 10218353 Ki = 1290 nM T03500 C1C7AH 10223757 Ki > 5025 nM T03500 CV5X8A 10224181 IC50 > 30000 nM T03500 CGKU70 10224396 Ki = 370 nM T03500 CO8M7Q 10239526 Ki > 6020 nM T03500 CEO4X5 10239762 Ki > 6020 nM T03500 CU7TQ3 10239803 Ki > 6020 nM T03500 CBM0Y4 10252411 Ki < 100 nM T03500 CGP97S 10274748 Ki = 520 nM T03500 CR48SA 10289842 Ki = 1030 nM T03500 CO60CU 10290029 Ki = 4100 nM T03500 CDU36Y 10296475 Ki = 338.84 nM T03500 C48IRP 10296785 Ki = 320 nM T03500 CE1KM9 10311498 Ki = 580 nM T03500 CJ15OB 10311501 Ki > 6020 nM T03500 C5F0EV 10311947 Ki > 6020 nM T03500 C7G6QW 10312268 Ki > 6020 nM T03500 CQ5IT9 10312372 Ki = 4640 nM T03500 CQY4C7 10318433 IC50 = 100 nM T03500 CIDW49 10319098 Ki > 6023 nM T03500 CJWH74 10321975 Ki > 6023 nM T03500 CI0T8K 10366352 Ki > 6023 nM T03500 C6WZ4F 10367355 IC50 = 57 nM T03500 CSY8C1 10387791 IC50 = 400 nM T03500 CFKA79 10395015 Ki = 2000 nM T03500 CN1K2Y 10408590 IC50 = 460 nM T03500 C5WV1N 10439082 Ki > 2000 nM T03500 CX38EB 10467565 IC50 > 100000 nM T03500 C9XC8Y 10493383 IC50 = 42 nM T03500 CG32FM 10613145 IC50 = 9 nM T03500 CI4SQ2 10732349 IC50 > 100000 nM T03500 C3UCL2 10854279 IC50 = 13 nM T03500 C9WPH7 11016072 Ki = 380 nM T03500 CBE68H 11016073 Ki = 346.74 nM T03500 CR4V2D 11101785 Ki = 109.65 nM T03500 C43ONW 11202395 Ki > 6023 nM T03500 CU80AR 11213937 IC50 = 24 nM T03500 C1IW7N 11292680 IC50 = 0.2 nM T03500 C8C5AV 11294179 IC50 = 8000 nM T03500 COT41H 11305534 IC50 = 200 nM T03500 C48JVH 11327633 IC50 = 180 nM T03500 CJ5SU9 11328354 Ki > 300000 nM T03500 C49CDU 11335940 IC50 = 62 nM T03500 CHLQ56 11352067 IC50 = 7 nM T03500 C9ABX8 11397130 Ki > 6023 nM T03500 C7WPC3 11442210 IC50 = 13 nM T03500 CB3LS1 11475677 IC50 = 8300 nM T03500 C1OT2G 11487618 IC50 = 140 nM T03500 CJ46KN 11508259 Ki = 8 nM T03500 CI8R5J 11529867 IC50 = 25740 nM T03500 CE01PG 11543178 IC50 = 24690 nM T03500 CXT05D 11581283 IC50 = 320 nM T03500 CX2PQ5 11588332 IC50 = 7560 nM T03500 CZO71U 11639846 IC50 = 200 nM T03500 CNY92D 11640694 Ki = 9000 nM T03500 CR2UN0 11669859 IC50 = 2 nM T03500 C90GCV 11675055 IC50 = 600 nM T03500 C3U6ZR 11697504 Ki > 50000 nM T03500 C4FU2H 11717997 IC50 = 1140 nM T03500 CCD93H 11730086 Ki = 200 nM T03500 CO8QT0 11753905 Ki = 12 nM T03500 C02BWA 11967143 Ki = 35 nM T03500 CB80OT 12000718 IC50 = 655 nM T03500 C43PJZ 12000720 IC50 > 20000 nM T03500 C4R2DA 23645953 Ki > 300000 nM T03500 CWN3I4 23645959 Ki > 300000 nM T03500 CFK5V8 23661684 IC50 = 10400 nM T03500 C7KF1N 23729138 IC50 = 4 nM T03500 C3TWS6 24178109 Ki = 31 nM T03500 CXEP14 24754176 IC50 = 5600 nM T03500 CSQ9E4 24754248 IC50 = 1700 nM T03500 CX16GL 24754251 IC50 > 22000 nM T03500 COY8K0 24754252 IC50 > 22000 nM T03500 CY6KA0 24755074 IC50 = 46000 nM T03500 CUS47E 24795059 IC50 = 0.4 nM T03500 C18FRG 24807817 IC50 > 100000 nM T03500 CAZ95J 24857924 IC50 = 18 nM T03500 C4UEM5 24871537 Ki > 50000 nM T03500 CP2L5B 24871655 Ki > 50000 nM T03500 C78OAU 24944977 IC50 = 40 nM T03500 CO6CJ5 24945161 IC50 = 3500 nM T03500 C1C0NX 24945244 IC50 = 3300 nM T03500 CLTQ28 24945246 IC50 = 250 nM T03500 C7ZA6S 24945247 IC50 = 600 nM T03500 CB94KU 24958549 IC50 = 25000 nM T03500 CAQ9Z1 25022681 Ki > 6023 nM T03500 CA86UE 25049752 Ki = 6 nM T03500 C82NLV 25049754 Ki = 40 nM T03500 C6QFV4 25049756 Ki = 62 nM T03500 C4HVF2 25064051 IC50 = 10.3 nM T03500 C64BZH 25064052 IC50 = 1.8 nM T03500 CZ2TG0 25064053 IC50 = 50 nM T03500 C3S8OA 25064054 IC50 = 60 nM T03500 CA64KF 25064283 IC50 = 187 nM T03500 C94MXR 25064485 IC50 = 34.1 nM T03500 CD9T2O 25064489 IC50 = 260 nM T03500 C3BC9Z 25064704 IC50 = 1470 nM T03500 C23TDS 25064904 IC50 = 9 nM T03500 C54MLN 25064905 IC50 = 6.3 nM T03500 C7T2UO 25064906 IC50 = 20.2 nM T03500 C16AIC 25064907 IC50 = 29 nM T03500 CL9N8I 25064908 IC50 = 23.1 nM T03500 CJP30U 25065108 IC50 = 36.3 nM T03500 CMZV31 25065109 IC50 = 28 nM T03500 C03NHX 25065111 IC50 = 6.1 nM T03500 CE72DR 25065318 IC50 = 7.2 nM T03500 CEK1Y2 25065514 IC50 = 14 nM T03500 C3F5LH 25065515 IC50 = 39 nM T03500 CB0Z5P 25065946 IC50 = 11 nM T03500 CJWD41 25066149 IC50 = 170 nM T03500 CI4A7E 25066153 IC50 = 100 nM T03500 CN9UM1 25066154 IC50 = 7300 nM T03500 CEU95V 25066364 IC50 = 2900 nM T03500 C0FJK5 25066365 IC50 = 2100 nM T03500 CZY4L8 25066366 IC50 = 4400 nM T03500 C2ZS5J 25066563 IC50 = 6.2 nM T03500 C6CMU0 25066564 IC50 = 6.6 nM T03500 CZO08G 25066566 IC50 = 14 nM T03500 C58KNZ 25066763 IC50 = 2.1 nM T03500 CVR52U 25066764 IC50 = 2 nM T03500 C8IBO5 25066765 IC50 = 5.6 nM T03500 CP85RV 25067176 IC50 = 7.6 nM T03500 CXP6V8 25067178 IC50 = 1.1 nM T03500 C8IO9U 25117549 IC50 = 0.4 nM T03500 CE9WR8 25120748 IC50 = 17 nM T03500 C3DHI1 25121089 IC50 = 4.5 nM T03500 C17SZR 25121093 IC50 = 2.9 nM T03500 C26JLO 25122164 IC50 = 0.3 nM T03500 CRU03Q 25122901 IC50 = 0.1 nM T03500 C6N7EQ 25138258 Ki = 160 nM T03500 C7AD1J 25138259 Ki = 70 nM T03500 CJ9TQ2 25138260 Ki = 65 nM T03500 CUT8I7 25138261 Ki = 107 nM T03500 CBD9X6 25138262 Ki = 53 nM T03500 C8LX1S 25138263 Ki = 43 nM T03500 C3OV1L 25138264 Ki = 85 nM T03500 C92WVM 25138265 Ki = 10 nM T03500 CMCS41 25138266 Ki = 1021 nM T03500 C1FJV5 25138267 Ki = 580 nM T03500 C9N6WT 25138268 Ki = 540 nM T03500 CF4QI1 25138269 Ki = 3245 nM T03500 C6P5UL 25138270 Ki = 327 nM T03500 CQE0L7 25138271 Ki = 119 nM T03500 C59XWU 25138272 Ki = 160 nM T03500 CR35QP 25144971 IC50 > 5000 nM T03500 C0Y5BC 25145683 IC50 > 2500 nM T03500 CHR2P1 25183768 Ki > 25000 nM T03500 C8IM5D 25263230 IC50 = 50 nM T03500 C7PTR2 25263231 IC50 = 2500 nM T03500 C9MR1P 25263232 IC50 = 70 nM T03500 CW9MK2 25263233 IC50 = 45 nM T03500 CX9L6V 25263234 IC50 = 1050 nM T03500 CJE4M1 25263235 IC50 = 3900 nM T03500 CJ1H5A 25263236 IC50 = 5 nM T03500 C2CGD1 25263237 IC50 = 4.7 nM T03500 C57UXR 25263238 IC50 = 10.2 nM T03500 CO4K7N 25263239 IC50 = 5 nM T03500 C3TGE2 25263240 IC50 = 0.9 nM T03500 C06WRU 25263241 IC50 = 12 nM T03500 C95AVW 25263242 IC50 = 10 nM T03500 CXT42G 25263243 IC50 = 16 nM T03500 C50DHY 25263244 IC50 = 38 nM T03500 C6R7SI 25263245 IC50 = 600 nM T03500 C9GCO4 28602444 IC50 > 150000 nM T03500 CCI64J 44224245 IC50 = 1.4 nM T03500 CLRT69 44247751 IC50 = 0.2 nM T03500 CX4VZ8 44248449 IC50 = 7.6 nM T03500 C3JP6F 44248450 IC50 = 25 nM T03500 CD94XA 44248451 IC50 > 1000 nM T03500 C90ZLT 44248570 IC50 = 18 nM T03500 CF8G2N 44248571 IC50 = 89 nM T03500 CSY0M2 44248572 IC50 = 44 nM T03500 CHM1D7 44248573 IC50 = 17 nM T03500 CM3Y8J 44248697 IC50 = 42 nM T03500 CF49LH 44248698 IC50 = 100.1 nM T03500 CCXS75 44248811 IC50 = 9.2 nM T03500 CUSR91 44248815 IC50 = 11.1 nM T03500 CH48TD 44315155 IC50 = 93 nM T03500 C62FXJ 44315244 IC50 = 1.698 nM T03500 C50IQE 44315333 IC50 = 3.981 nM T03500 CGQ92A 44364037 IC50 = 72 nM T03500 C36YLM 44364111 IC50 = 191 nM T03500 CN4T7Q 44364119 IC50 = 59 nM T03500 CH4TE7 44364121 IC50 = 57 nM T03500 CPE91Y 44364122 IC50 = 29 nM T03500 CG2X0C 44364224 IC50 = 421 nM T03500 C1F8XN 44364249 IC50 = 20 nM T03500 CWM47H 44364250 IC50 = 65 nM T03500 C0W5TL 44364251 IC50 = 931 nM T03500 C3TPO7 44364266 IC50 = 170 nM T03500 CJ2B8F 44364280 IC50 = 7689 nM T03500 CAF3O9 44389199 IC50 = 400 nM T03500 CF8NZ7 44389227 IC50 = 400 nM T03500 C0S7EU 44389231 IC50 = 70 nM T03500 CE9R5S 44389246 IC50 = 57 nM T03500 CN8F1Q 44389253 IC50 = 70 nM T03500 CB71LT 44389285 IC50 = 14 nM T03500 CC7QW9 44391352 IC50 = 29 nM T03500 CXD05N 44394645 Ki > 300000 nM T03500 CGQ98X 44394681 Ki = 49000 nM T03500 C8MY4S 44394703 Ki > 300000 nM T03500 CCEI41 44394814 Ki > 2000000 nM T03500 CCZ09V 44394886 Ki > 100000 nM T03500 CZB81D 44395506 IC50 < 1 nM T03500 CZ41FN 44426071 IC50 > 100000 nM T03500 C05OPT 44426072 IC50 > 100000 nM T03500 C45WZX 44426073 IC50 > 100000 nM T03500 C95DYN 44426074 IC50 > 100000 nM T03500 C8CJ4U 44426075 IC50 = 56900 nM T03500 C1K7QR 44426076 IC50 > 100000 nM T03500 CR7MF4 44426077 IC50 > 100000 nM T03500 C4GE1C 44426078 IC50 = 43600 nM T03500 CJN1K9 44439853 Ki = 50 nM T03500 CV58YW 44441018 Ki > 6023 nM T03500 CV85PN 44441019 Ki = 3560 nM T03500 C5O2WK 44441020 Ki > 6023 nM T03500 CU67WS 44441021 Ki > 6023 nM T03500 CXZ53B 44441022 Ki > 6023 nM T03500 C8S7UT 44441023 Ki > 6023 nM T03500 CT4PZ9 44441024 Ki > 6023 nM T03500 CU9GE6 44441025 Ki > 6023 nM T03500 CB2IT4 44441026 Ki > 6023 nM T03500 CN4X2F 44441027 Ki > 6023 nM T03500 CPF45Y 44441028 Ki > 6023 nM T03500 CAM23N 44441029 Ki > 6023 nM T03500 C23BPG 44441030 Ki = 958 nM T03500 C5YMT6 44441031 Ki > 6023 nM T03500 C9A6GJ 44441032 Ki > 6023 nM T03500 CYSU19 44441033 Ki > 6023 nM T03500 C0HX1L 44445199 IC50 = 67000 nM T03500 CPQT35 44445200 IC50 = 51000 nM T03500 C2X6IP 44445201 IC50 = 67000 nM T03500 CSRB79 44445202 IC50 = 71000 nM T03500 C2O6KZ 44445203 IC50 = 71000 nM T03500 CASF34 44445204 IC50 = 69000 nM T03500 CQZ6M0 44445205 IC50 = 68000 nM T03500 CH7Z5M 44445206 IC50 = 69000 nM T03500 C71CPO 44445207 IC50 = 82000 nM T03500 CO9QA4 44445209 IC50 = 69000 nM T03500 CH3UQ5 44445210 IC50 = 105000 nM T03500 C6B4LG 44445211 IC50 = 79000 nM T03500 C1WA5N 44445212 IC50 = 82000 nM T03500 CM2CD0 44445213 IC50 = 68000 nM T03500 C6ZX2P 44445214 IC50 = 16000 nM T03500 C9KE8P 44445215 IC50 = 65000 nM T03500 C68QEF 44445216 IC50 = 60000 nM T03500 CCK7W2 44445217 IC50 = 100000 nM T03500 C58BQA 44445218 IC50 = 20000 nM T03500 C4CGN2 44445219 IC50 = 31000 nM T03500 C1IVR6 44445220 IC50 = 56000 nM T03500 CG2U7H 44445221 IC50 = 63000 nM T03500 CVW48J 44445222 IC50 = 68000 nM T03500 CL3HZ8 44445223 IC50 = 47000 nM T03500 CPY73U 44445224 IC50 = 44000 nM T03500 C9MA2F 44445225 IC50 = 31000 nM T03500 C9SJM3 44445226 IC50 = 105000 nM T03500 CH91WG 44445228 IC50 = 70000 nM T03500 CO59HI 44445229 IC50 = 111000 nM T03500 C62WPE 44445230 IC50 = 97000 nM T03500 COIR35 44445231 IC50 = 105000 nM T03500 CBH0M7 44445233 IC50 = 99000 nM T03500 CIS7M5 44445234 IC50 = 118000 nM T03500 CKN60A 44445235 IC50 = 65000 nM T03500 CP4XL8 44445237 IC50 = 62000 nM T03500 CJA79R 44445239 IC50 = 76000 nM T03500 CA72BI 44445240 IC50 = 68000 nM T03500 CZJB48 44445241 IC50 = 146000 nM T03500 C85EVH 44445242 IC50 > 150000 nM T03500 C9DI7F 44445243 IC50 = 87000 nM T03500 CVLH67 44445244 IC50 = 82000 nM T03500 CIP3X8 44445245 IC50 = 117000 nM T03500 CL1MK6 44445246 IC50 = 85000 nM T03500 C0CX7T 44445247 IC50 = 70000 nM T03500 CEZ2P7 44445248 IC50 = 81000 nM T03500 CL0K9Q 44445249 IC50 = 134000 nM T03500 C9T2SH 44445250 IC50 = 94000 nM T03500 C5EFP9 44445251 IC50 = 78000 nM T03500 CLJ71G 44445252 IC50 = 96000 nM T03500 C8TF3E 44445253 IC50 = 78000 nM T03500 C4CAY7 44445254 IC50 = 151000 nM T03500 CH1LE5 44445255 IC50 = 112000 nM T03500 CLP96W 44445256 IC50 = 127000 nM T03500 CK8S4Z 44445257 IC50 = 17000 nM T03500 C03EJW 44445258 IC50 = 106000 nM T03500 CO9SM5 44445261 IC50 = 115000 nM T03500 C3FX8B 44445262 IC50 > 150000 nM T03500 CZS8N5 44445263 IC50 > 150000 nM T03500 CMW2U6 44445264 IC50 = 101000 nM T03500 CB47AH 44445265 IC50 = 135000 nM T03500 CA43LS 44445266 IC50 = 52000 nM T03500 C23MDF 44445267 IC50 = 71000 nM T03500 C9K3DI 44445268 IC50 = 109000 nM T03500 C2ZAK4 44445269 IC50 = 93000 nM T03500 CIVC64 44445270 IC50 = 105000 nM T03500 C8W1HX 44445271 IC50 > 150000 nM T03500 CTFR27 44445272 IC50 > 150000 nM T03500 C20DNO 44445273 IC50 > 150000 nM T03500 CWLC15 44445274 IC50 > 150000 nM T03500 CZD5M3 44445275 IC50 > 150000 nM T03500 CJET46 44445276 IC50 > 150000 nM T03500 CI58AM 44445277 IC50 = 61000 nM T03500 CDN37V 44445278 IC50 > 150000 nM T03500 CE36AB 44445279 IC50 > 150000 nM T03500 CV9KX5 44445280 IC50 > 150000 nM T03500 C4S2WX 44445281 IC50 > 150000 nM T03500 CG0Z7I 44478924 IC50 = 920 nM T03500 CFO27Y 44478926 IC50 = 32 nM T03500 CBZJ29 44478927 IC50 = 4.8 nM T03500 CRJ24K 44479197 IC50 = 2.7 nM T03500 CGOH82 44479198 IC50 = 380 nM T03500 CLV56M 44479199 IC50 = 140 nM T03500 CY92OQ 44479458 IC50 = 5800 nM T03500 CH1QG9 44479459 IC50 = 70 nM T03500 CB1NT7 44479460 IC50 = 6 nM T03500 C0JQ9L 44479699 IC50 = 6 nM T03500 C0DN1Q 44479700 IC50 = 89000 nM T03500 CTG24W 44479702 IC50 = 1900 nM T03500 CGZ49M 44479703 IC50 = 310 nM T03500 CPA8F4 44555417 IC50 = 1240 nM T03500 CUE6Z1 44555419 IC50 = 2020 nM T03500 C10SGK 44555421 IC50 = 2990 nM T03500 CK68GT 44580539 Ki = 29.5 nM T03500 C0KR6J 44626353 IC50 = 58 nM T03500 C25QLI 44626354 IC50 = 55 nM T03500 C2HI5Q 45269910 IC50 = 87 nM T03500 C84JSF 45269911 IC50 = 750 nM T03500 CMPE63 45482676 IC50 = 410 nM T03500 CGH1U8 45482997 IC50 = 181 nM T03500 C8AUI5 45482999 IC50 = 54400 nM T03500 C9W7IP 45483016 IC50 = 1150 nM T03500 CPB42K 45483022 IC50 = 20100 nM T03500 CBG76X 45483023 IC50 = 19900 nM T03500 CDW4C8 45483036 IC50 = 3750 nM T03500 CY8N4A 45485460 IC50 > 100000 nM T03500 CH9DL7 45485461 IC50 > 100000 nM T03500 CN3L8A 45485463 IC50 > 100000 nM T03500 CZ2H8A 45485476 IC50 > 100000 nM T03500 CS2CF0 45485477 IC50 > 100000 nM T03500 C48SNP 45485482 IC50 = 5020 nM T03500 CN7C6O 45485485 IC50 > 100000 nM T03500 CI1DY0 45485486 IC50 > 100000 nM T03500 C0KB7R 45485487 IC50 > 100000 nM T03500 CJ5W7S 45485502 IC50 > 100000 nM T03500 C02NQW 45485508 IC50 > 100000 nM T03500 CAM9T0 45485513 IC50 > 100000 nM T03500 C6FE2C 45485514 IC50 = 5020 nM T03500 CZ3Q6V 45485515 IC50 = 18700 nM T03500 C8G3MA 45485520 IC50 > 100000 nM T03500 C0WP1Z 45485521 IC50 > 100000 nM T03500 CL8Q3B 45485532 IC50 = 10200 nM T03500 CV8FP3 45485558 IC50 > 100000 nM T03500 C56WVI 46184724 Ki = 700 nM T03500 CL2U4Z 46829322 Ki = 7.6 nM T03500 C0F7SU 46905989 IC50 = 64000 nM T03500 C2S7PK 46942365 Ki = 14.3 nM T03500 C7XW1Q 50907084 Ki = 7 nM T03500 C8RL5Q 50907292 Ki = 60 nM T03500 CU2SX3 51355576 Ki = 1350 nM T03500 CRI92N 53311230 IC50 > 10000 nM T03500 C91ERL 53318212 IC50 = 85 nM T03500 CWH47R 53319228 Ki = 11 nM T03500 CM96EW 53320529 IC50 = 3600 nM T03500 C29OHB 53326114 IC50 = 31000 nM T03500 C6Y2EV 53374826 IC50 > 100000 nM T03500 CJH01K 54580192 IC50 = 70 nM T03500 C6R3MZ 54580973 Ki > 50000 nM T03500 CWKA42 54582019 Ki = 2300 nM T03500 CO3WV0 54582221 IC50 = 90 nM T03500 C62FZC 56835063 IC50 = 1 nM T03500 CKJ9S1 56835167 IC50 = 23 nM T03500 C21CLZ 56835168 IC50 = 19 nM T03500 C0L2TS 56835169 IC50 = 66 nM T03500 CQU16V 57339411 Ki = 23 nM T03500 C6LM3B 57339412 Ki = 16 nM T03500 CNVG85 57339413 Ki = 10 nM T03500 CHE2I1 57345500 Ki > 50000 nM T03500 C63TFM 57345501 Ki > 50000 nM T03500 C8KT2F 57345502 Ki = 12000 nM T03500 C0KPD8 57384084 IC50 = 2500 nM T03500 CV67JB 57384091 IC50 = 500 nM T03500 C80XPO 57390510 IC50 = 0.2 nM T03500 CA9Q8Z 57390511 IC50 < 1 nM T03500 C6GBO2 57390512 IC50 = 1.2 nM T03500 C3F1XQ 57390513 IC50 = 1.6 nM T03500 CDN25L 57390514 IC50 = 4 nM T03500 CN2H9K 57391204 IC50 > 10000 nM T03500 CR8MW2 57391205 IC50 > 10000 nM T03500 C74TRW 57392282 IC50 = 18 nM T03500 C4NAD0 57392283 IC50 = 0.2 nM T03500 CNQ9B2 57392969 IC50 > 100000 nM T03500 CTYP14 57392972 IC50 > 10000 nM T03500 C5VB0U 57392973 IC50 > 10000 nM T03500 CMQL31 57392974 IC50 > 10000 nM T03500 C39OHF 57392975 IC50 > 10000 nM T03500 CB5NV1 57394039 IC50 = 1.9 nM T03500 CNOH63 57394711 IC50 = 7943.28 nM T03500 CS01IU 57395798 IC50 = 7.2 nM T03500 C7BD4V 57397577 IC50 = 0.7 nM T03500 CW5DB1 57397578 IC50 = 2.2 nM T03500 C39MHB 57397579 IC50 = 5.4 nM T03500 CP1L0G 57399258 IC50 = 0.4 nM T03500 CH01LU 57399259 IC50 = 2.2 nM T03500 CL61FT 57399260 IC50 = 2.3 nM T03500 CD50CO 57399918 IC50 > 10000 nM T03500 C1PW0D 57401025 IC50 = 23 nM T03500 CXGN63 57401026 IC50 = 8.6 nM T03500 CL49YN 57402781 IC50 = 13 nM T03500 CUYR63 57402782 IC50 = 15 nM T03500 CK68EY 57403424 IC50 > 10000 nM T03500 C0G2VY 57403564 IC50 = 19 nM T03500 C6BKQ0 57874709 IC50 = 2100 nM T03500 C8ITK7 59794408 IC50 = 3.3 nM T03500 CSO3W8 59794423 IC50 = 23.7 nM T03500 C6JE9N 59794437 IC50 = 8.9 nM T03500 C7ECU2 59794447 IC50 = 5.9 nM T03500 CAT67H 59910477 IC50 = 295.8 nM T03500 CHP8D4 66560535 IC50 = 13000 nM T03500 CH95AD 66560623 IC50 = 48000 nM T03500 C8B6WD 70688393 IC50 = 670 nM T03500 C6P3XM 70693710 Ki > 50000 nM T03500 C0HE2P 70694634 IC50 = 1790 nM T03500 CU90BG 70698422 Ki = 0.28 nM T03500 C1HVB4 70698423 Ki = 15.5 nM T03500 C2C7SA 71563039 Ki = 14.7 nM T03500 CH5J4A 71602247 IC50 = 44 nM T03500 CH53IU 71602248 IC50 = 400 nM T03500 C97EWQ 71602249 IC50 = 500 nM T03500 CYS46I 71652677 IC50 = 2100 nM T03500 CX67VE 71654516 IC50 = 2300 nM T03500 C72HNL 71720757 IC50 = 0.93 nM T03500 CKV2U5 71817094 Ki = 10 nM T03500 CHDS52 71817095 Ki = 5 nM T03500 C5LZH0 71817097 Ki = 2 nM T03500 C50SID 71817098 Ki = 15 nM T03500 CN83DB 71817100 Ki = 6 nM T03500 CW5IQ0 73345859 Ki = 9 nM T03500 CW01EA 73349535 IC50 > 100000 nM T03500 C43WKX 73353429 Ki = 1 nM T03500 CK42DO 73353430 Ki = 7 nM T03500 C6H5TU 73354941 Ki = 5 nM T03500 C06BPT 73355130 IC50 = 2 nM T03500 CEHB08 73356503 Ki = 272 nM T03500 CA5T7P 73603957 IC50 = 26 nM T03500 C8VN1R 74221194 IC50 = 9 nM T03500 C8ID2O 76314808 Ki = 1 nM T03500 C01TZS 76325699 Ki = 48 nM T03500 CE09XI 76332924 Ki = 3.53 nM T03500 CUE7G4 86287514 IC50 = 70 nM T03500 CAB2F5 87349434 Ki = 270 nM T03500 CO2FL5 90137145 IC50 = 5 nM T03500 C4OD0K 118225789 IC50 = 10000 nM T03500 CDO15M 118721026 IC50 = 138 nM T03500 CQ6C8V 121232412 IC50 = 18 nM T03500 C89QOM 127043503 IC50 = 462 nM T03500 C9E5YJ 127043505 IC50 = 63 nM T03500 CW1Q3D 127043506 IC50 = 84 nM T03500 C1C7WB 127044036 IC50 = 296.6 nM T03500 CPF6U7 127044139 IC50 = 177.6 nM T03500 CT9B0Q 127044462 IC50 = 71.02 nM T03500 CL3X1A 127044649 IC50 = 246.6 nM T03500 C8RZ7T 127044651 IC50 = 52.3 nM T03500 C3I4PT 127044652 IC50 = 96.1 nM T03500 CDX86T 127044818 IC50 = 73.2 nM T03500 C56OJV 127044819 IC50 = 53.2 nM T03500 CYA92R 130282633 IC50 = 13 nM T03500 CO3QE2 130282636 IC50 = 6 nM T03500 C83FAY 134130294 Ki = 23 nM T03500 C1MOD4 135567320 IC50 = 467 nM T03500 CL9Y5Q 135678161 IC50 > 10000 nM T03500 CA5JR6 136054481 IC50 = 300 nM T03500 CV47JN 136054485 IC50 = 260 nM T03500 CZ48WO 136054487 IC50 = 9500 nM T03500 C8FGT0 136054495 IC50 = 540 nM T03500 CG70BZ 136054516 IC50 = 8.5 nM T03500 CSM57W 136054520 IC50 = 1.8 nM T03500 CXNG40 136118011 Ki = 4120 nM T03500 C1IOH9 136118012 Ki = 3611 nM T03500 CTY79S 136118013 Ki > 5025 nM T03500 CTE87J 136118014 Ki > 5025 nM T03500 CIEW62 136380958 IC50 = 16 nM T03500 C9HS7J 137287436 IC50 = 8.1 nM T03500 CB8M6U 137646865 IC50 = 1800 nM T03500 CS80YI 137652598 IC50 = 7 nM T03500 CAB7Q6 137660566 IC50 = 930 nM T03500 CZ8H6N 137661550 IC50 = 9 nM T03500 C6IPV3 145949783 IC50 = 493250 nM T03500 C72LGN 145950074 IC50 > 500000 nM T03500 CBA49I 145955092 IC50 = 54.7 nM T03500 C2HAG8 145955226 IC50 > 500000 nM T03500 COR96H 145956298 IC50 = 493200 nM T03500 C7R3FE 145956426 IC50 = 100100 nM T03500 CQ15DP 145957734 IC50 = 198300 nM T03500 CG03OE 145959777 IC50 = 95200 nM T03500 CIQ9J2 145960035 IC50 = 109100 nM T03500 CJ9B6C 145963868 IC50 = 1250 nM T03500 C42AZM 145965977 IC50 = 200 nM T03500 C8M7FR 145966330 IC50 = 26 nM T03500 C5ICD0 145967022 IC50 = 510 nM T03500 C8DF3N 145967770 IC50 = 4000 nM T03500 C72NJI 145968012 IC50 = 297 nM T03500 CRK13Q 145969600 IC50 = 11 nM T03500 CWY5X0 145971805 IC50 = 40 nM T03500 CN73DF 145972870 IC50 = 8.5 nM T03500 CYFI60 145973042 IC50 = 7500 nM T03500 C3F0AD 145973196 IC50 = 502 nM T03500 CZ2XC4 145973252 IC50 > 10000 nM T03500 CI9VB4 145975902 IC50 > 10000 nM T03500 C1KPL5 145976497 IC50 = 33 nM T03500 CZ4SB5 145976911 IC50 > 10000 nM T03500 C18OCA 145976989 IC50 = 230000 nM T03500 C6T9CX 145979814 IC50 = 40000 nM T03500 CK1A9G 145979968 IC50 = 9600 nM T03500 CFP7Q1 145979987 IC50 = 19 nM T03500 CB2J6O 145980521 IC50 = 1300 nM T03500 CLK6W4 145980984 IC50 = 65 nM T03500 C0OV4I 145982041 IC50 = 98 nM T03500 C6ZTV3 145986744 IC50 = 9200 nM T03500 CX15IY 145986836 IC50 = 83 nM T03500 C1TSJ5 145987118 IC50 = 51 nM T03500 CC82EI 145987827 IC50 = 20 nM T03500 CNR3F4 145991781 IC50 = 41 nM T03500 C89PNI 145992859 IC50 = 40 nM T03500 CT7BR3 145994093 IC50 = 84 nM T03500 C3XL6T 155510956 Ki = 0.9 nM T03500 CF64GH 155518335 Ki = 1340 nM T03500 CJN8X5 155542058 Ki = 1 nM T03500 CC3G0X 155561622 Ki = 0.26 nM T03500 CLT4Y6 10138589 Ki = 280 nM T03500 D02ECA 448942 IC50 = 14 nM T03500 D04UBY 45483018 IC50 = 3390 nM T03500 D04VPH 45376872 IC50 > 22000 nM T03500 D05JPV 44406790 IC50 = 12480 nM T03500 D05THD 44478925 IC50 = 590 nM T03500 D06EHW 11625778 IC50 = 17 nM T03500 D07MJD 44479701 IC50 = 1500 nM T03500 D08ELY 9838786 IC50 = 12 nM T03500 D09MLQ 25122902 IC50 = 0.1 nM T03500 D09ZOA 25049753 Ki = 2 nM T03500 D0A0FY 44479457 IC50 = 14000 nM T03500 D0A5MV 11581319 IC50 = 450 nM T03500 D0B3UN 44580458 Ki = 0.19 nM T03500 D0C1EQ 20348772 IC50 = 11800 nM T03500 D0F4UT 21496278 IC50 = 4500 nM T03500 D0G3YZ 11391583 IC50 = 340 nM T03500 D0K0YX 44626352 IC50 = 86 nM T03500 D0L4EO 11609208 IC50 = 480 nM T03500 D0L6ND 10089677 IC50 = 0.33 ug.mL-1 T03500 D0LB0N 45483008 IC50 = 7840 nM T03500 D0LM2K 45483015 IC50 = 2490 nM T03500 D0N6CD 10565532 IC50 = 14 nM T03500 D0S9OL 10155934 IC50 = 1200 nM T03500 D0T1FR 44457233 IC50 > 100000 nM T03500 D0TL3N 45482998 IC50 = 3530 nM T03500 D0XK7G 10445302 Ki = 20 nM T03500 D0Y5IQ 44255320 IC50 = 5000 nM T03500 D0YN1A 893637 IC50 = 290 nM T72545 D0O1WX 2764 IC50 = 51000 nM T72545 D0IY0R 11591505 IC50 = 2200 nM T72545 CECV23 11604842 IC50 = 16 ug.mL-1 T72545 CX9QP0 11837127 IC50 = 4100 nM T72545 CD07QM 44403289 IC50 = 27.8 ug.mL-1 T72545 CQ7MB8 121415395 IC50 = 900 nM T72545 C1G2WE 121415404 IC50 = 10000 nM T72545 C5IU4C 121415407 IC50 = 2500 nM T72545 C1H8UD 121415415 IC50 = 200 nM T72545 CG9O1K 121415456 IC50 = 59000 nM T72545 CI51CM 121415469 IC50 = 2400 nM T72545 CB2VC9 121415490 IC50 = 100 nM T72545 CCN1U2 121415509 IC50 = 100 nM T72545 CCT46D 121415540 IC50 = 100 nM T72545 CBL05X 121417642 IC50 = 2200 nM T72545 CE87PY 121417653 IC50 = 7300 nM T72545 CN9T8M 121417654 IC50 = 3100 nM T72545 CZ7XB1 121417677 IC50 = 22600 nM T72545 CSH51T 121417711 IC50 = 130000 nM T72545 C2IRX6 121417737 IC50 = 28500 nM T72545 C6OP3Z 121418109 IC50 = 22900 nM T72545 CH08PV 121429867 IC50 = 1700 nM T72545 C3FW9K 121433130 IC50 = 700 nM T72545 CX6F2R 135462833 IC50 = 13.9 ug.mL-1 T72545 C57TMP 155511431 IC50 = 2400 nM T72545 CUZ0M6 155522161 IC50 = 29300 nM T72545 CAJ91F 155531127 IC50 = 1300 nM T72545 C09COM 155532384 IC50 = 1300 nM T72545 C4V7UR 155538148 IC50 = 52500 nM T72545 CXJ1G9 155544331 IC50 = 3800 nM T72545 C7UDQ2 155545881 IC50 = 400 nM T72545 CLB2V4 155546018 IC50 = 13100 nM T72545 C79USC 155548113 IC50 = 1100 nM T72545 CG4E8A 155548135 IC50 = 1900 nM T72545 CED32V 155549037 IC50 = 3200 nM T72545 CIR6C4 155549058 IC50 = 7800 nM T72545 CQ7T6H 155549145 IC50 = 6700 nM T72545 C06ZCE 155556229 IC50 = 1700 nM T72545 CZUE35 155558181 IC50 = 1200 nM T72545 CIW64O 155560768 IC50 = 900 nM T72545 CXW42N 155563849 IC50 = 8000 nM T72545 C9E5MU 155566312 IC50 = 8800 nM T72545 CQYI40 155568240 IC50 = 3900 nM T55956 D00AXJ 4189 IC50 = 6500 nM T55956 D00ENY 33032 EC50 = 4900 nM T55956 D02VKC 3272524 IC50 = 74000 nM T55956 D0D4OW 57338826 IC50 = 3300 nM T55956 D0U5CS 213056 EC50 = 2990 nM T55956 COC91V 10255 EC50 = 299000 nM T55956 C8NO0Z 77937 EC50 > 1000000 nM T55956 C9H6OS 92136 EC50 = 140000 nM T55956 CUBH61 101122 EC50 > 1000000 nM T55956 CB15YI 125799 EC50 > 1000000 nM T55956 CLMU31 165627 EC50 > 1000000 nM T55956 C34YGT 173564 EC50 > 1000000 nM T55956 CF2EW1 308248 IC50 = 71000 nM T55956 CJOQ02 674768 IC50 = 750 nM T55956 C2Z6CA 921213 IC50 = 4100 nM T55956 C5F8YH 2733519 IC50 > 300000 nM T55956 CZ1Q5P 4694355 Ki > 1000000 nM T55956 C05WNA 5310956 Ki = 5800 nM T55956 CRL5Z4 5353536 IC50 = 23000 nM T55956 C3RTI9 6348408 EC50 = 6700 nM T55956 C9INH1 6604707 EC50 > 1000000 nM T55956 CD68LI 6604795 Ki = 58000 nM T55956 C9PJQ1 9794208 IC50 = 1380 nM T55956 C9XQK6 10198133 EC50 = 2430 nM T55956 CX12HM 10330132 Ki > 1000000 nM T55956 C3KHU7 10465017 EC50 > 1000000 nM T55956 CH9VN3 10560963 EC50 > 1000000 nM T55956 CDN69Z 10609381 EC50 > 1000000 nM T55956 C8CH1R 10684992 IC50 = 8600 nM T55956 CQTF38 10775369 EC50 = 800000 nM T55956 C9BK1A 10846649 EC50 = 5300 nM T55956 CDO7A1 10979251 EC50 = 1270 nM T55956 CJ5B8P 11084869 IC50 = 3040 nM T55956 C8LSU6 11275666 EC50 = 9370 nM T55956 CL1VX3 11310142 EC50 = 7540 nM T55956 CX2T1N 11344646 EC50 = 9280 nM T55956 CP9Y7Q 15479143 EC50 = 1410 nM T55956 CJS57V 16061421 EC50 = 6100 nM T55956 C6Q4GL 16747847 EC50 = 1950 nM T55956 CM7JD0 16747848 EC50 = 3410 nM T55956 CWU3X9 16748099 EC50 = 111000 nM T55956 CI9FL7 24779948 EC50 > 100000 nM T55956 CJR05E 24780088 EC50 = 31000 nM T55956 C5OQ7F 24780092 EC50 > 100000 nM T55956 C7F4YL 24780225 EC50 = 30000 nM T55956 C7E8SH 44322745 Ki > 1000000 nM T55956 CGL0Z3 44322843 Ki > 1000000 nM T55956 C2SKJ1 44322921 Ki = 5300 nM T55956 CHV03D 44338561 EC50 = 410000 nM T55956 C96FCM 44817555 IC50 = 3500 nM T55956 CVF45M 44817558 IC50 = 10000 nM T55956 CKCT65 44817595 IC50 = 12000 nM T55956 C6J8WQ 44817596 IC50 = 5700 nM T55956 CZR5N0 44817597 IC50 = 2400 nM T55956 C3FXD0 44817625 IC50 = 3600 nM T55956 C0O4BI 44817627 IC50 = 10600 nM T55956 CFX4P2 44817688 IC50 = 21000 nM T55956 CY94XB 45483692 IC50 = 38000 nM T55956 CO6AH4 45483698 IC50 = 54000 nM T55956 CKB74O 46918013 EC50 = 8800 nM T55956 C1VY4Z 46918015 EC50 = 6000 nM T55956 C0L2SP 51036108 EC50 > 30000 nM T55956 CAU6D5 51036701 EC50 > 30000 nM T55956 CBI3A0 51036916 EC50 > 30000 nM T55956 C3GQ8O 51037131 EC50 > 30000 nM T55956 CE4KP1 51050257 Ki > 10000 nM T55956 CY58NO 53240406 EC50 = 3450 nM T55956 CJRG27 54761054 EC50 > 30000 nM T55956 CZ0A1T 57765525 EC50 = 4000 nM T55956 C49IAZ 57765535 EC50 = 18000 nM T55956 C4BZ0U 57765536 EC50 = 4600 nM T55956 C9QDZ0 57765549 EC50 > 100000 nM T55956 CSI9E0 57765613 EC50 = 4000 nM T55956 CBFD61 57765616 EC50 = 2900 nM T55956 CC82HD 57765622 EC50 = 5700 nM T55956 CQ70WE 57765633 EC50 = 4200 nM T55956 CISA81 58058356 EC50 = 26000 nM T55956 CPDW56 58058372 EC50 = 3200 nM T55956 CQY10C 58058380 EC50 > 100000 nM T55956 C8JAU2 60096211 EC50 = 709 nM T55956 C8N4UB 60096231 EC50 = 1950 nM T55956 C4PU9N 67056056 EC50 > 30000 nM T55956 CCT07V 68290289 EC50 > 10000 nM T55956 C03JUE 68290572 EC50 > 10000 nM T55956 CZT05A 69929646 EC50 > 30000 nM T55956 CG7F5Z 70051296 EC50 = 6690 nM T55956 CBK2Y6 70051926 IC50 = 267 nM T55956 CZ6XT7 70052526 EC50 = 4370 nM T55956 CNIW83 71479388 EC50 > 30000 nM T55956 C8U0CT 71681823 EC50 = 780 nM T55956 CO5P1V 71681824 EC50 = 11800 nM T55956 C6EIO9 71681825 IC50 = 1890 nM T55956 CLH9N3 71681826 EC50 = 3250 nM T55956 C0VN8X 92044496 EC50 = 3600 nM T55956 CUC13P 122187795 IC50 > 30000 nM T55956 CCP5U2 122195692 EC50 > 10000 nM T55956 CH2AO4 122539788 IC50 > 30000 nM T55956 C2MEI0 124425164 EC50 = 2400 nM T55956 CPZ70S 127052897 EC50 > 30000 nM T55956 C38BRY 131801162 EC50 > 10000 nM T55956 CFC05Q 131954513 EC50 > 10000 nM T55956 C3EGM5 137321168 IC50 > 10000 nM T55956 CS7O0A 137634883 EC50 = 4500 nM T55956 C9H6NY 137639752 EC50 = 3600 nM T55956 CK2W6L 137640190 EC50 = 2400 nM T55956 CAI63F 137642874 EC50 = 3200 nM T55956 CS5F0B 137644345 EC50 = 23000 nM T55956 C9U6EI 137645989 EC50 = 1100 nM T55956 CCW58E 137646034 EC50 > 100000 nM T55956 C3PDO0 137647077 EC50 = 3900 nM T55956 CO9L1G 137650519 EC50 = 1070 nM T55956 CT1M7B 137654697 EC50 = 68400 nM T55956 CMQ61F 137655963 EC50 = 10200 nM T55956 CDWR37 137661492 EC50 > 100000 nM T55956 C9C8KU 137661528 EC50 = 760 nM T55956 C3IL9H 155511336 IC50 > 30000 nM T55956 CYXE53 155538270 IC50 > 10000 nM T55956 CZ7NH0 155545491 IC50 > 30000 nM T55956 D00IGI 2207 EC50 = 280 nM T55956 D04DKM 104766 Ki = 60000 nM T55956 D05TFE 5218788 Ki > 100000 nM T55956 D06DUE 40539 Ki = 1000000 nM T55956 D06PAK 10058694 Ki = 2400 nM T55956 D07GRG 10197984 Ki = 400 nM T55956 D08CAB 83887 EC50 > 1000000 nM T55956 D09AQK 4545574 Ki = 4700 nM T55956 D09QUN 58368068 EC50 > 10000 nM T55956 D09RPR 16737207 Ki > 10000 nM T55956 D0B2VW 95883 IC50 = 4000 nM T55956 D0D2GL 3972752 Ki = 480000 nM T55956 D0EK6P 5310984 Ki = 110000 nM T55956 D0IO8J 3025961 Ki > 10000 nM T55956 D0KL4K 71041983 EC50 = 4200 nM T55956 D0L0YF 4236420 EC50 = 82000 nM T55956 D0LC5O 16062593 EC50 = 3200 nM T55956 D0N0NJ 15508178 Ki = 20000 nM T55956 D0O1AK 23327 EC50 > 1000000 nM T55956 D0OT9B 5960 EC50 > 1000000 nM T55956 D0PN6Z 179394 EC50 = 55 nM T55956 D0Q6VH 5311432 Ki > 100000 nM T55956 D0T5SU 158397 EC50 = 220000 nM T55956 D0V2VU 3997004 IC50 = 4500 nM T55956 D0W3PY 6604820 EC50 = 11000 nM T39519 D0N1XD 6223 IC50 = 260 nM T39519 CU54KV 3084126 IC50 = 530 nM T39519 CQS5Z1 10417379 IC50 = 66 nM T39519 CBX8T9 16451230 IC50 > 150000 nM T39519 C6QZM4 46885506 IC50 > 10000 nM T39519 C02ORV 53377508 Ki > 20000 nM T39519 CPL71I 54596764 IC50 > 100000 nM T39519 C72GHW 56642706 IC50 > 100000 nM T39519 CS6Q7R 56642708 IC50 > 100000 nM T39519 CV8A4S 56676725 IC50 = 1100 nM T39519 CJBY70 56951879 Ki > 50000 nM T39519 CER5F1 67466175 IC50 > 100000 nM T39519 C8JTS3 70676140 Ki > 100000 nM T39519 CZL47S 70676141 Ki > 100000 nM T39519 C8KC6O 70676142 Ki > 100000 nM T39519 CUP4Q6 76328021 Ki > 50000 nM T39519 CX7V5M 76328022 Ki > 50000 nM T39519 C5P2BM 76331683 Ki > 50000 nM T39519 D02TVQ 71268957 IC50 > 100000 nM T39519 D04FNI 11657687 IC50 = 800 nM T39519 D09CLP 439155 IC50 = 1200 nM T07930 D0E3SH 6918837 Ki = 0.7 nM T07930 D0E7PQ 5311 Ki = 33 nM T07930 D0L7LC 5352062 Ki = 550 nM T07930 D0Y3KG 3121 IC50 > 2000000 nM T07930 D00FHR 9865515 IC50 > 10000 nM T07930 D05KED 53340666 IC50 = 5000 nM T07930 D06TKI 49857317 IC50 = 200 nM T07930 D07FPY 6918877 Ki = 17 nM T07930 D09XIZ 11538455 Ki = 2.1 nM T07930 D0B1FE 3194 IC50 = 3400 nM T07930 D0B3FV 6445533 IC50 = 5.58 nM T07930 D0B7CH 4775 IC50 > 2000000 nM T07930 D0E6UZ 54575456 IC50 = 406 nM T07930 D0GE5B 56654642 IC50 > 180000 nM T07930 D0GH3Q 9804992 Ki = 600 nM T07930 D0L2UQ 49855250 Ki = 21 nM T07930 D0M8FD 4261 IC50 = 1400 nM T07930 D0XT6W 6918638 Ki = 25 nM T07930 D0Z4RC 24756910 IC50 = 11.4 nM T07930 D0J8OC 5186 IC50 = 300 nM T07930 D00HXJ 118884610 Ki = 701 nM T07930 D0L1NO 72722126 IC50 = 10 nM T07930 D0QX3G 71532921 IC50 > 10000 nM T07930 D0YN2T 86302836 IC50 = 16 nM T07930 D0N3SH 4996 Ki = 4750 nM T07930 CBIR94 10313 IC50 > 33330 nM T07930 C1N2KZ 88129 IC50 = 37000 nM T07930 C35INR 338818 IC50 = 1270 nM T07930 CH1JD3 419176 IC50 = 360000 nM T07930 C0Y4WC 614947 Ki > 2500 nM T07930 CU3HS2 1108280 IC50 > 100000 nM T07930 C18ENP 6918846 Ki = 18 nM T07930 C1RD7E 6918878 IC50 > 10000 nM T07930 CE9LP2 9543539 IC50 > 180000 nM T07930 CJ84NF 9815304 IC50 > 10000 nM T07930 CC0EU7 9828788 IC50 > 10000 nM T07930 C7RC1E 10309899 IC50 = 7.1 nM T07930 CG9L1R 10435243 IC50 = 1308 nM T07930 C60QVT 10460379 IC50 = 3040 nM T07930 C9OU5F 10464879 Ki > 2500 nM T07930 CDY91S 10584105 Ki > 2500 nM T07930 CSMT47 10728039 Ki > 2500 nM T07930 CK8UV7 11019840 Ki > 2500 nM T07930 CRZ7H2 11556677 IC50 > 10000 nM T07930 CQ32FV 11664499 IC50 = 2500 nM T07930 CG9OC4 11682502 IC50 = 21.8 nM T07930 CYB26W 11688197 IC50 > 1000 nM T07930 CC3GQ0 11700059 IC50 > 10000 nM T07930 C9G1BN 11993595 IC50 = 4900 nM T07930 CH5JS7 11993694 IC50 = 311 nM T07930 CJ94OC 12542182 Ki > 2500 nM T07930 CXJ5G9 13190582 IC50 > 10000 nM T07930 C06UTF 13507024 IC50 = 1600 nM T07930 C1KR4L 14113324 IC50 > 50000 nM T07930 C15MQN 14113325 IC50 = 21000 nM T07930 C2D1KP 15983982 Ki = 9.2 nM T07930 CHB82E 15986417 IC50 = 78400 nM T07930 C52EVH 15986418 IC50 = 11200 nM T07930 CS1QO9 15986509 IC50 = 29600 nM T07930 CQGC05 16036765 IC50 = 1900 nM T07930 CM3T2E 16049824 IC50 > 1 nM T07930 CFK8J5 16068056 Ki = 11 nM T07930 CMQP70 16068495 Ki = 11 nM T07930 CT84XO 16068594 Ki = 6.6 nM T07930 CF3ZG5 16068595 Ki = 6.8 nM T07930 CL60CA 16068912 Ki = 5.6 nM T07930 C5CIB4 16663079 IC50 > 50000 nM T07930 CWO7V0 16733295 IC50 = 310 nM T07930 CV54SY 16733414 IC50 = 890 nM T07930 C8RC9P 24744325 IC50 > 50000 nM T07930 C17GDO 24779722 IC50 = 134 nM T07930 CIO7Q6 24853792 IC50 > 10000 nM T07930 CBN0J5 24853793 IC50 > 10000 nM T07930 CV8EF6 25032862 IC50 > 50000 nM T07930 CX69SY 25066355 IC50 = 1340 nM T07930 CF8VP4 25066356 IC50 = 878 nM T07930 CS9XH7 25066547 IC50 = 695 nM T07930 C46AGN 25066548 IC50 = 55.4 nM T07930 CJF2M7 25066549 IC50 = 341 nM T07930 C4I1CJ 25155417 IC50 > 50000 nM T07930 CB4E2J 25155956 IC50 > 50000 nM T07930 CO14XG 25195084 IC50 > 10000 nM T07930 CCD5M7 25227504 IC50 = 62.2 nM T07930 CK0D5S 25227505 IC50 = 155 nM T07930 CN97JP 25227508 IC50 = 109 nM T07930 CW8R1B 25227513 IC50 = 150 nM T07930 C43BHY 25269097 IC50 = 354 nM T07930 C2KO0F 42599456 IC50 = 7.6 nM T07930 C1UAO7 42601485 IC50 > 50000 nM T07930 CDT65Y 42631047 IC50 > 100000 nM T07930 CO57GS 44138033 IC50 = 3670 nM T07930 C5VP4D 44454144 IC50 > 50000 nM T07930 CJ0L4C 44456965 IC50 = 1900 nM T07930 C7F8YJ 44543715 Ki = 11500 nM T07930 CEM91G 44562802 IC50 = 10 nM T07930 CIO34V 44564642 Ki = 16 nM T07930 CA6Q9Y 44592060 IC50 = 10800 nM T07930 C5H8RA 44598536 IC50 > 10000 nM T07930 CC2QV9 44623002 IC50 > 50000 nM T07930 CVJ51M 44623152 IC50 > 50000 nM T07930 C6TJ2G 44623153 IC50 > 50000 nM T07930 CO7S9W 44626297 IC50 = 110 nM T07930 CSM1O6 45271073 IC50 = 28000 nM T07930 C96ROY 45482635 IC50 > 10000 nM T07930 CV74KP 45482658 IC50 > 10000 nM T07930 CHC0Y1 45482667 IC50 = 470 nM T07930 C69UBY 46861822 IC50 = 31000 nM T07930 C8D4XL 46861823 IC50 = 31000 nM T07930 CPSI47 46890583 Ki = 13 nM T07930 C90NYX 46896338 IC50 = 3500 nM T07930 CL7PS1 49831258 IC50 > 50000 nM T07930 CI5L2P 49846123 IC50 = 38540.65 nM T07930 C4DL0M 49847150 IC50 = 1930 nM T07930 CC7Y9U 49850262 IC50 = 2300 nM T07930 C50PXU 49855444 IC50 > 50000 nM T07930 C6POK9 49856931 IC50 = 500 nM T07930 C78GKN 53361474 IC50 = 892 nM T07930 CNB63X 53361475 IC50 = 932 nM T07930 CQ43VH 53363518 Ki = 3.1 nM T07930 C6Y2EV 53374826 IC50 = 34700 nM T07930 CYQV72 54030066 IC50 = 150 nM T07930 C5A7MU 54613496 IC50 = 2.5 nM T07930 CIO96M 56659403 IC50 > 100000 nM T07930 CL18NI 56666337 IC50 > 100000 nM T07930 C9LC5Y 56673234 IC50 > 100000 nM T07930 CWH5N4 56673261 IC50 > 100000 nM T07930 CCW89V 56932477 IC50 = 850 nM T07930 CZ25SN 56935695 IC50 > 30000 nM T07930 C41ZBJ 56951446 Ki > 50000 nM T07930 C1R7HZ 56951447 Ki = 13000 nM T07930 CP4EL2 57328394 IC50 = 15000 nM T07930 C60XUA 57336554 Ki > 50000 nM T07930 C58USD 57336555 Ki > 50000 nM T07930 C4DZ0B 57336556 Ki > 50000 nM T07930 C7JCL9 57336558 Ki > 50000 nM T07930 CN9W2G 57336559 Ki > 50000 nM T07930 C10DMC 57336560 Ki > 50000 nM T07930 CLR1C6 57336561 Ki > 50000 nM T07930 CU6B5H 57336562 Ki > 50000 nM T07930 CWTK67 57336564 Ki > 50000 nM T07930 C95REB 57336565 Ki > 50000 nM T07930 CU68CZ 57336566 Ki > 50000 nM T07930 C0JQ2U 57336567 Ki > 50000 nM T07930 C8O0CH 57336568 Ki > 50000 nM T07930 C5CN3K 57336569 Ki > 50000 nM T07930 CO0RD1 57336570 Ki > 50000 nM T07930 CDK61Y 57336571 Ki > 50000 nM T07930 C0BT1I 57336572 Ki > 50000 nM T07930 C8ZBR3 57401090 Ki > 50000 nM T07930 C4LI0D 57521296 IC50 = 9 nM T07930 CA5Q6O 58147189 IC50 > 50000 nM T07930 C4DYC0 58147224 IC50 > 50000 nM T07930 CMP04X 58147302 IC50 > 50000 nM T07930 CLD40J 58465708 IC50 = 29000 nM T07930 C1MB4Q 59323957 IC50 > 30000 nM T07930 CK6LX0 59454220 IC50 = 5300 nM T07930 C2SDN1 59454252 IC50 = 1100 nM T07930 CO6A2S 59585196 IC50 = 35000 nM T07930 CPZ5Q3 60148646 IC50 = 150 nM T07930 CP2HK9 60148667 IC50 = 30 nM T07930 C8ZL3J 60148690 IC50 = 9 nM T07930 CK5N4E 60148693 IC50 = 4 nM T07930 C27DKW 60148711 IC50 = 30 nM T07930 CS2E6C 60148712 IC50 = 50 nM T07930 CPF50R 60148997 IC50 = 340 nM T07930 CB7X2E 60151224 IC50 > 10000 nM T07930 CY05OU 60151225 IC50 > 10000 nM T07930 CWO8H0 60152596 IC50 > 10000 nM T07930 CBN3L0 69950064 Ki = 182 nM T07930 CQY1I6 70789579 Ki = 24300 nM T07930 C0CX7P 71476624 Ki > 2500 nM T07930 C6QPH1 71476625 Ki > 2500 nM T07930 C3JLD4 71476626 Ki > 2500 nM T07930 C3OH6T 71476627 Ki > 2500 nM T07930 C0LWJ6 71520631 IC50 = 2.31 nM T07930 CO28HI 71520716 IC50 = 33.4 nM T07930 CVA5Q7 71520717 IC50 = 4.22 nM T07930 C89SWX 71527724 IC50 > 30000 nM T07930 CKR6U8 71583101 IC50 = 1800 nM T07930 CBZ5S9 71583103 IC50 = 500 nM T07930 C3PSJ9 71583105 IC50 = 500 nM T07930 C7HG0K 71655802 IC50 = 18320 nM T07930 CPJ4V7 71680913 IC50 > 33000 nM T07930 CI9G3B 71681069 IC50 = 26000 nM T07930 CIR56T 71721558 IC50 > 100000 nM T07930 CCD18W 71721946 IC50 > 100000 nM T07930 CFUC24 71722010 IC50 > 10000 nM T07930 CT7L6G 72163687 Ki > 2500 nM T07930 CKE9D3 72163688 Ki > 2500 nM T07930 CI9H6L 72164895 IC50 = 3891 nM T07930 CV09DJ 72734543 IC50 > 10000 nM T07930 CX3W1T 73333311 IC50 = 3300 nM T07930 CM6H9C 76324878 IC50 = 7 nM T07930 CKI74A 76853213 IC50 > 20000 nM T07930 CJ6Z0X 78324068 IC50 > 20000 nM T07930 C3U0KE 81689842 IC50 = 60 nM T07930 C61VCD 86294741 IC50 = 37000 nM T07930 CBWV30 86294747 IC50 = 27000 nM T07930 C06YBD 86302594 IC50 = 1580 nM T07930 C6M9PL 86765212 IC50 = 8730 nM T07930 CS5I4Y 87261507 IC50 = 220 nM T07930 CYW51P 90654946 IC50 = 124000 nM T07930 CJH1S6 90654947 IC50 > 100000 nM T07930 CSR56C 90655296 IC50 = 1910 nM T07930 CSDO81 90664458 Ki = 21 nM T07930 CJO6T1 91810840 IC50 = 9500 nM T07930 C34WIG 92045024 IC50 > 100000 nM T07930 C9OC0F 101882265 IC50 = 36000 nM T07930 CT7Z8F 102514716 IC50 = 26570 nM T07930 CSU52M 118656852 IC50 = 1300 nM T07930 CB6AJ9 118656853 IC50 = 400 nM T07930 C1JFZ7 118714371 IC50 = 9850 nM T07930 C2M5OR 118714376 IC50 = 3540 nM T07930 CI8G4X 118737400 IC50 = 9370 nM T07930 CB84TO 121278998 IC50 = 20000 nM T07930 C9S5OK 121279020 IC50 > 50000 nM T07930 CL3M2F 121499152 IC50 > 33330 nM T07930 C28JVO 122192004 IC50 > 10000 nM T07930 CF2D8U 122192005 IC50 > 10000 nM T07930 C3V5ND 122550211 IC50 > 10000 nM T07930 CZE35C 122648343 IC50 > 1000 nM T07930 C54RNT 122648367 IC50 = 750 nM T07930 C1UVI7 122648600 IC50 > 1000 nM T07930 CMX59K 122648648 IC50 = 484 nM T07930 CVZ64I 122648649 IC50 > 1000 nM T07930 CV9I8D 127030313 IC50 = 8000 nM T07930 CB8HR2 129104138 IC50 = 39000 nM T07930 CCH65A 129104183 IC50 > 50000 nM T07930 CFH8Q4 129104227 IC50 > 50000 nM T07930 C6HM5P 129104349 IC50 > 50000 nM T07930 CZTF90 129104374 IC50 > 50000 nM T07930 CUJ2P5 129104402 IC50 > 50000 nM T07930 CY3I6X 129104426 IC50 = 18000 nM T07930 C6X3HG 132145728 IC50 = 2251 nM T07930 C8O9DP 132157820 IC50 = 3112 nM T07930 C4KE3N 132938351 IC50 = 5391 nM T07930 C05FVT 134492522 IC50 > 10000 nM T07930 C14FWK 135348858 IC50 = 6910 nM T07930 CS1V6A 135367138 IC50 > 50000 nM T07930 CVO59N 135367789 IC50 > 50000 nM T07930 CDY18W 135407493 IC50 > 100000 nM T07930 CW2I4R 135412048 IC50 > 100000 nM T07930 C7U0AV 135412194 IC50 > 100000 nM T07930 CS54TL 135437514 IC50 > 100000 nM T07930 C36MUC 135441620 IC50 > 100000 nM T07930 CRB8M1 135444536 IC50 > 100000 nM T07930 CX5D6J 135446479 IC50 = 27900 nM T07930 C1TOK2 135449197 IC50 > 100000 nM T07930 CW25GL 135462117 IC50 > 100000 nM T07930 CCL28F 135473106 IC50 > 100000 nM T07930 CYA60G 135497781 IC50 = 94300 nM T07930 C8X5LO 135928012 Ki = 180 nM T07930 CI2YE8 135928628 IC50 > 100000 nM T07930 C50NIS 136025837 IC50 > 100000 nM T07930 C4OS0V 136025842 IC50 > 100000 nM T07930 CX7Z5B 136025843 IC50 > 100000 nM T07930 CB8EM9 136025984 IC50 > 100000 nM T07930 C49MUG 136025986 IC50 > 100000 nM T07930 CH7Y3C 136086920 IC50 > 100000 nM T07930 C3VDL5 136086921 IC50 > 100000 nM T07930 C9GOB5 136086922 IC50 = 48600 nM T07930 CE3ZL7 136086923 IC50 > 100000 nM T07930 CJZ5F3 136086924 IC50 = 16700 nM T07930 CT19ND 136110961 IC50 > 100000 nM T07930 CY9U0E 136173089 IC50 > 50000 nM T07930 CRPN39 136645466 IC50 > 10000 nM T07930 C67EFJ 137628684 IC50 > 1000 nM T07930 CP0BN3 137631704 Ki > 50000 nM T07930 CPOF51 137632251 Ki > 50000 nM T07930 CZ1FK2 137635119 IC50 > 50000 nM T07930 C6JVG9 137635398 IC50 = 10500 nM T07930 C8GNS5 137645287 IC50 = 356000 nM T07930 CGMN16 137647616 Ki > 50000 nM T07930 CDXE54 137649646 Ki > 50000 nM T07930 C5FHD3 137652442 IC50 = 200 nM T07930 CB15PI 137652670 Ki > 50000 nM T07930 CCR5B3 137654793 IC50 = 7400 nM T07930 C1SBN5 137654946 IC50 = 1030 nM T07930 CI6R3W 137656303 Ki > 50000 nM T07930 C76OGQ 137656942 IC50 = 9100 nM T07930 C1DL3P 137657892 Ki > 50000 nM T07930 C8D2GT 137658785 Ki > 50000 nM T07930 CAQ62X 137701235 Ki = 360 nM T07930 CN2UH1 139303146 IC50 = 16740 nM T07930 C7XI0V 141764754 IC50 = 540 nM T07930 CX0E9B 142505968 IC50 = 43700 nM T07930 C9G5ZW 142505990 IC50 = 100000 nM T07930 C7N8LV 142506025 IC50 = 9087 nM T07930 CKBF56 142506033 IC50 = 23610 nM T07930 CLND62 142506170 IC50 = 10000 nM T07930 CGNQ74 142506189 IC50 = 2144 nM T07930 C1T3IQ 142506210 IC50 = 8106 nM T07930 CP5HF8 142506225 IC50 = 3827 nM T07930 CDA28I 145949712 IC50 = 16840 nM T07930 CV3QO5 145951170 IC50 > 10000 nM T07930 CKG98W 145953085 IC50 > 100000 nM T07930 CL0XT8 145954248 IC50 = 2967 nM T07930 C9IV1C 145959866 IC50 > 10000 nM T07930 CK1XI0 145960971 IC50 > 10000 nM T07930 CP53JS 145977717 IC50 > 10000 nM T07930 CWD0A9 145983712 Ki = 1000 nM T07930 C56MWZ 145986208 Ki = 4200 nM T07930 C0GMR1 146585718 IC50 = 439 nM T07930 C0YXS8 147254231 IC50 = 1356 nM T07930 CN71OS 149405396 IC50 = 8592 nM T07930 C8S3MF 150076000 IC50 > 300 nM T07930 C9FIY4 153534005 IC50 > 10000 nM T07930 CQ5BL7 155512551 IC50 > 50000 nM T07930 CE4H7I 155513471 IC50 > 50000 nM T07930 CW3VT9 155514603 IC50 > 50000 nM T07930 CZ84WI 155515284 IC50 > 50000 nM T07930 CUKG21 155515602 IC50 > 50000 nM T07930 CYJ53T 155515864 IC50 = 8000 nM T07930 CA1J3N 155517086 IC50 = 4600 nM T07930 CL72ME 155517175 IC50 > 10000 nM T07930 CY54TU 155518062 IC50 = 400 nM T07930 CEH2N5 155518106 IC50 = 14900 nM T07930 CAD06U 155519254 IC50 = 3120 nM T07930 CDY5H6 155519645 IC50 = 5510 nM T07930 CAZ3S7 155521187 IC50 = 22000 nM T07930 CZ75FW 155521272 IC50 = 4600 nM T07930 CZ70PO 155529066 IC50 > 50000 nM T07930 C49NGT 155529137 IC50 > 50000 nM T07930 CN3W5J 155531452 IC50 = 34000 nM T07930 CK2UY4 155531957 IC50 = 2700 nM T07930 CIZ46A 155533876 IC50 = 12000 nM T07930 C6LB5D 155535084 IC50 = 27000 nM T07930 CTF98X 155537473 IC50 = 5300 nM T07930 CAG9P4 155537573 IC50 = 4000 nM T07930 CLD19W 155539311 IC50 = 7860 nM T07930 CU6V4Q 155539319 IC50 > 50000 nM T07930 C6U0FM 155540189 IC50 = 6800 nM T07930 CP4L1F 155544459 IC50 > 50000 nM T07930 CXR86J 155545078 IC50 > 50000 nM T07930 CF2O4J 155546325 IC50 > 50000 nM T07930 CS3GO2 155546558 IC50 = 3400 nM T07930 C0AU1L 155546632 IC50 > 50000 nM T07930 C90FBZ 155549087 IC50 > 50000 nM T07930 C4Z5JX 155550827 IC50 > 50000 nM T07930 CGDF76 155554360 IC50 = 9100 nM T07930 C7QTU1 155555957 IC50 > 50000 nM T07930 CGL24S 155562249 IC50 = 16100 nM T07930 CPNA06 155564750 IC50 > 50000 nM T07930 CZDC03 155565491 IC50 > 30000 nM T07930 CG65CR 155565674 IC50 > 50000 nM T07930 CD05RS 155566122 IC50 = 50000 nM T07930 C4A0RK 155566461 IC50 > 50000 nM T07930 C04CGS 155567444 IC50 > 50000 nM T07930 CS03PJ 155568350 IC50 = 9500 nM T07930 D00GBB 11449246 Ki = 46 nM T07930 D01YBR 44591988 IC50 = 7360 nM T07930 D02NWS 279980 Ki = 16000 nM T07930 D03BQS 45482666 IC50 = 1460 nM T07930 D03QOD 239512 IC50 = 140 nM T07930 D04KQF 6675804 Ki = 1500 nM T07930 D04UVL 1133083 IC50 > 50000 nM T07930 D05OVV 11993691 IC50 = 590 nM T07930 D06IMY 44626296 IC50 = 110 nM T07930 D07YZZ 5173 Ki = 9500 nM T07930 D09RKA 72946782 IC50 = 5000 nM T07930 D0A4HF 45482630 IC50 = 90 nM T07930 D0E0TA 44454650 IC50 > 50000 nM T07930 D0E9DD 16095101 IC50 = 10000 nM T07930 D0FN5D 45482672 IC50 = 280 nM T07930 D0H4YW 3611 Ki > 2500 nM T07930 D0I4RK 45482660 IC50 = 1200 nM T07930 D0K7QR 45269423 IC50 = 140 nM T07930 D0M9LJ 44454415 IC50 > 50000 nM T07930 D0MD7H 44454143 IC50 > 50000 nM T07930 D0N9AK 44138031 IC50 = 7200 nM T07930 D0PK9V 45482643 IC50 = 210 nM T07930 D0Q2GM 44454416 IC50 > 50000 nM T07930 D0Q5DI 71462653 IC50 = 6620 nM T07930 D0R7JA 53344908 IC50 = 80 nM T07930 D0T0SK 44138032 IC50 = 1160 nM T07930 D0T4JQ 264 IC50 > 2000000 nM T07930 D0U8FC 759408 IC50 > 50000 nM T07930 D0Z8PX 24757913 IC50 > 10000 nM T95438 D00ENY 33032 IC50 = 52000 nM T95438 C9CQV1 131738 IC50 = 240000 nM T95438 C45TML 1755783 IC50 > 300000 nM T95438 CDK9W5 1796705 IC50 > 300000 nM T95438 C8L6JU 2177697 IC50 > 300000 nM T95438 CRQW20 2266743 IC50 > 300000 nM T95438 CO0I2U 2266913 IC50 > 300000 nM T95438 C9HE6N 2271641 IC50 > 300000 nM T95438 CH4RP6 2271698 IC50 > 300000 nM T95438 C3SL4Y 2271738 IC50 > 300000 nM T95438 C7K9MX 2283576 IC50 > 300000 nM T95438 CB6EZ4 2285406 IC50 > 300000 nM T95438 CBW36C 2287441 IC50 > 300000 nM T95438 C13DLB 2289587 IC50 > 300000 nM T95438 CZQ83G 2289624 IC50 > 300000 nM T95438 CFG35Z 2737891 IC50 > 100000 nM T95438 CYR4X2 2838960 IC50 > 100000 nM T95438 CP4L3M 2839392 IC50 > 300000 nM T95438 CF2LE3 4133412 IC50 = 1995.26 nM T95438 CP2RL5 5310957 IC50 = 4000 nM T95438 CJW9P4 5506801 IC50 > 300000 nM T95438 C5PWJ3 6505351 IC50 > 300000 nM T95438 CTBZ42 6505352 IC50 > 300000 nM T95438 CV2J5T 6604785 Ki = 1600 nM T95438 C64QSY 7016554 Ki = 32359.37 nM T95438 CTMP80 9920506 Ki = 10715.19 nM T95438 C2EA8S 10219727 IC50 = 490000 nM T95438 C53YBE 10419887 Ki > 400000 nM T95438 C2PE4O 10464763 IC50 = 300000 nM T95438 C46KUE 10680281 Ki = 67608.3 nM T95438 C9V6WM 10866618 Ki = 12000 nM T95438 C2WQB7 10877814 IC50 > 1000000 nM T95438 C83OPZ 10954230 IC50 > 1000000 nM T95438 C7Z6AX 10986716 IC50 = 430000 nM T95438 C78YAI 10997729 IC50 > 1000000 nM T95438 CE80SU 11041159 IC50 > 1000000 nM T95438 CMSD95 11062853 IC50 > 1000000 nM T95438 C2TWR9 11063103 IC50 > 1000000 nM T95438 C0HT8M 11528550 Ki = 21877.62 nM T95438 CQ5H1B 11543205 Ki = 52000 nM T95438 C2QJU5 11616374 IC50 = 100 nM T95438 CZ9V5S 11629898 Ki = 21877.62 nM T95438 C5E8BT 11651356 Ki = 38018.94 nM T95438 CV76LO 11667702 IC50 = 100 nM T95438 C7SHB1 11745400 Ki = 20892.96 nM T95438 C0BM2Z 12047098 IC50 = 2000 nM T95438 C68AOJ 12047099 IC50 = 1300 nM T95438 C09XIT 12047100 IC50 = 2200 nM T95438 C1X3YB 16727662 IC50 > 300000 nM T95438 C6XLF5 24905646 Ki = 290000 nM T95438 CFI54P 24905647 Ki = 630957.34 nM T95438 CQK96U 24905648 Ki = 1000000 nM T95438 C36NMZ 24905649 IC50 = 300000 nM T95438 CB3T7C 24905650 IC50 = 75000 nM T95438 C14RNW 24905651 Ki = 125892.54 nM T95438 CM1S2B 24905652 Ki = 290000 nM T95438 CUS45D 24905703 IC50 > 3000000 nM T95438 C86BUK 24905705 IC50 = 3000000 nM T95438 CJ25EZ 44404580 IC50 = 200 nM T95438 C0LJ8T 44404590 IC50 = 500 nM T95438 CJD1V7 44404611 IC50 = 300 nM T95438 CJ6ER9 44404615 IC50 = 700 nM T95438 C4CZN1 44405320 Ki = 16218.1 nM T95438 CI94LS 44417413 Ki = 19952.62 nM T95438 C8TMX2 44417425 Ki = 6309.57 nM T95438 CR2IM7 49910175 IC50 > 300000 nM T95438 CY91US 52941382 IC50 = 17 nM T95438 CH5Z6U 52942568 IC50 = 21000 nM T95438 C2NK4G 52943726 IC50 = 25000 nM T95438 CEM8I5 52944933 IC50 = 14000 nM T95438 CHD72C 52945190 IC50 = 1400 nM T95438 CH6ZK2 52949825 IC50 = 19000 nM T95438 CVE68A 52949856 IC50 = 17000 nM T95438 C5ILP4 70682198 IC50 = 1300 nM T95438 C4HI0U 70789291 IC50 = 1000000 nM T95438 CP48NY 71449125 IC50 = 300 nM T95438 C7NYC0 71449126 IC50 = 200 nM T95438 CD03AH 71449127 IC50 = 100 nM T95438 CVST26 71450915 IC50 = 100 nM T95438 C31HCW 71450916 IC50 = 500 nM T95438 CC15SM 71450917 IC50 = 300 nM T95438 CBZ9D6 71450918 IC50 = 1000 nM T95438 CSO9P3 71452727 IC50 = 600 nM T95438 C23DMA 71452728 IC50 = 100 nM T95438 CE0A3V 71452729 IC50 = 700 nM T95438 CRKN62 71452730 IC50 = 130 nM T95438 C8X4VU 71454504 IC50 = 300 nM T95438 COUY80 71454505 IC50 <= 10 nM T95438 C8QW6K 71454506 IC50 = 400 nM T95438 CKWF24 71454507 IC50 = 1000 nM T95438 CDY5K2 71456248 IC50 = 200 nM T95438 C9O7LC 71456249 IC50 = 80 nM T95438 C1HJF2 71458054 IC50 = 200 nM T95438 C3P0MQ 71461655 IC50 = 13000 nM T95438 C0P4NT 71574743 IC50 > 300000 nM T95438 CGH79X 71574744 IC50 > 300000 nM T95438 COC8W2 71574746 IC50 > 300000 nM T95438 C5U9HZ 71574747 IC50 > 300000 nM T95438 C35BOJ 71574834 IC50 = 300000 nM T95438 CNVG02 71574836 IC50 = 300000 nM T95438 C2JS0I 71574837 IC50 = 24000 nM T95438 CV5IT8 71574838 IC50 = 700000 nM T95438 CL9BJ8 71574839 IC50 > 1000000 nM T95438 CCS4T2 71574840 IC50 > 1000000 nM T95438 CM5Z0I 71574841 IC50 > 300000 nM T95438 C3Z0TH 73348758 Ki = 6600 nM T95438 C8DGU5 90480101 IC50 > 1000000 nM T95438 CEH82V 90480134 IC50 > 1000000 nM T95438 CT2KF1 127030385 IC50 > 300000 nM T95438 CX95LC 127030386 IC50 > 300000 nM T95438 C8TS1X 127030387 IC50 > 300000 nM T95438 CF6NI8 127031290 IC50 > 300000 nM T95438 C2V5PM 132820245 IC50 = 84 nM T95438 CC54HS 134131748 IC50 = 50000 nM T95438 CM8O9I 134131963 IC50 = 1096.48 nM T95438 C26CTG 134132565 IC50 = 300000 nM T95438 CGXV98 134133631 IC50 = 7300 nM T95438 C1ZAB4 134134123 IC50 = 316227.77 nM T95438 CZ2WH5 134134813 IC50 = 30000 nM T95438 CT3MU6 134135313 IC50 = 50000 nM T95438 CTL6A4 134135682 IC50 = 60255.96 nM T95438 C0MJT1 134136786 IC50 = 2754.23 nM T95438 CA40DU 134137403 IC50 = 50000 nM T95438 C1L9UX 134139672 IC50 = 3300 nM T95438 CC24GI 134139698 IC50 = 501187.23 nM T95438 CTSA19 134139982 IC50 = 22000 nM T95438 CWS62H 134140412 IC50 = 43000 nM T95438 C5QIB1 134140490 IC50 = 10715.19 nM T95438 CT4QN8 134141720 IC50 = 6456.54 nM T95438 CJF5X7 134143016 IC50 = 70000 nM T95438 C4CT5L 134144465 IC50 = 6760.83 nM T95438 CL0EA9 134144947 IC50 = 100000 nM T95438 COM76W 134147363 IC50 > 300000 nM T95438 C9Q2JY 134147568 IC50 = 4677.35 nM T95438 CS38BI 134147884 IC50 = 2691.53 nM T95438 CP10YS 134148109 IC50 = 50000 nM T95438 CTPS85 134149212 IC50 = 6606.93 nM T95438 COP15G 134149427 IC50 = 500 nM T95438 C6HQS8 134149488 IC50 = 2398.83 nM T95438 CTH41F 134149576 IC50 = 25118.86 nM T95438 CQ8R9N 134149841 IC50 = 13489.63 nM T95438 C10RSO 134150446 IC50 > 300000 nM T95438 C9N0CQ 134152035 IC50 = 316227.77 nM T95438 C5SN8C 134152143 IC50 = 5000 nM T95438 C3RAO8 134153858 IC50 = 3235.94 nM T95438 CI3HS7 134155673 IC50 = 3019.95 nM T95438 CVT7Q4 134157558 IC50 = 4677.35 nM T95438 CHK48B 137643975 IC50 > 1000000 nM T95438 C6J8RH 137658224 IC50 > 1000000 nM T95438 CS1X0H 145952067 IC50 = 16.6 nM T95438 C2X6ST 145952092 IC50 = 690 nM T95438 CRXG02 145952717 IC50 = 1621.81 nM T95438 CZD62V 145953140 IC50 = 830 nM T95438 C5SH4V 145953224 IC50 = 81283.05 nM T95438 C63MDC 145954707 IC50 = 107.15 nM T95438 C87HDC 145955435 IC50 = 2754.23 nM T95438 CT3H6G 145955563 IC50 = 1584.89 nM T95438 CIN7D3 145955863 IC50 = 933.25 nM T95438 CZ7N3B 145956590 IC50 = 489.78 nM T95438 CFZK42 145957754 IC50 = 770 nM T95438 CEX81Q 145958688 IC50 = 74131.02 nM T95438 C6BP3Z 145959256 IC50 = 2400 nM T95438 C8DIJ6 145960111 IC50 = 1400 nM T95438 CET93L 145971223 IC50 = 18.2 nM T95438 CGF5S1 145971489 IC50 = 33000 nM T95438 C30JVP 145971753 IC50 = 758.58 nM T95438 CI04HT 145972021 IC50 = 46.77 nM T95438 C18GNB 145973375 IC50 = 36 nM T95438 CK7UW9 155519942 IC50 > 300000 nM T95438 C0Y9UF 155520160 IC50 > 300000 nM T95438 C52DFC 155524441 IC50 > 300000 nM T95438 C4IWE9 155525454 IC50 > 300000 nM T95438 CHJ5G1 155527881 IC50 > 300000 nM T95438 C9Z2ME 155529757 IC50 > 300000 nM T95438 CN1S4G 155530850 IC50 > 300000 nM T95438 C7HOI6 155533200 IC50 > 300000 nM T95438 CG65QS 155536541 IC50 > 300000 nM T95438 CX3ED4 155538143 IC50 > 300000 nM T95438 C4J3DC 155541203 IC50 > 300000 nM T95438 CD4B0V 155542542 IC50 > 300000 nM T95438 C87POT 155548017 IC50 > 300000 nM T95438 CPQM13 155555116 IC50 > 300000 nM T95438 CV9R4S 155557780 IC50 > 300000 nM T95438 C6NAQ5 155561202 IC50 > 300000 nM T95438 CF9YI6 155564787 IC50 > 300000 nM T95438 CFN45I 155565203 IC50 > 300000 nM T95438 CCK6T7 155565355 IC50 > 300000 nM T95438 D02JJX 11531745 IC50 = 70.79 nM T95438 D03RGP 1221 IC50 > 1000000 nM T95438 D03UIR 24905704 Ki = 158489.32 nM T95438 D04XZP 107883 IC50 = 79432.82 nM T95438 D07GUB 5311218 IC50 = 960 nM T95438 D09HET 11622683 IC50 = 42000 nM T95438 D0B2VW 95883 Ki = 11748.98 nM T95438 D0F5SO 11369932 IC50 = 700 nM T95438 D0JT2N 443239 IC50 = 9549.93 nM T95438 D0OT9B 5960 IC50 = 32000 nM T95438 D0X3CF 442879 IC50 > 100000 nM T11793 D00YZA 5453 Ki = 2200 nM T11793 D00YZD 54726191 IC50 > 100000 nM T11793 D04MSM 2554 EC50 = 145000 nM T11793 D05LBU 5472 Ki = 200 nM T11793 D06GKN 2099 IC50 < 10000 nM T11793 D06NXY 5991 Ki = 800 nM T11793 D07KSG 2733526 Ki = 900 nM T11793 D08QMX 5757 EC50 = 4100 nM T11793 D09KTS 24821094 IC50 = 11100 nM T11793 D09OJQ 4095 Ki = 10000 nM T11793 D0F9BY 166548 IC50 > 17500 nM T11793 D0G3DL 135398735 EC50 = 1300 nM T11793 D0H0HJ 19493 IC50 = 6200 nM T11793 D0K9MY 11243969 IC50 > 50000 nM T11793 D0N0TZ 60606 Ki = 500 nM T11793 D0N3VR 71616 Ki = 340 nM T11793 D0ZU9R 392622 IC50 = 2000 nM T11793 D03WNG 73051463 IC50 > 10000 nM T11793 D05LRD 59286554 IC50 > 30000 nM T11793 D06MHZ 66558287 IC50 = 5900 nM T11793 D06TQR 76287260 IC50 = 77000 nM T11793 D06ZEO 54674461 IC50 > 50000 nM T11793 D08AOZ 86582336 IC50 > 40000 nM T11793 D08VSQ 59336911 IC50 > 40000 nM T11793 D09DXX 71571306 IC50 > 100000 nM T11793 D0C9PZ 91754484 IC50 > 50000 nM T11793 D0DH5X 44472635 IC50 > 100000 nM T11793 D0G5XV 135565884 IC50 > 30000 nM T11793 D0I3LO 91933883 IC50 > 20000 nM T11793 D0N5KS 154104 IC50 < 10000 nM T11793 D0S5IR 86294073 IC50 > 30000 nM T11793 D0V9VG 51049968 IC50 >= 20000 nM T11793 D0YB2Y 42641863 Ki > 30000 nM T11793 D0QZ8K 70874141 IC50 = 61000 nM T11793 D04RLX 148201 IC50 > 100000 nM T11793 D09VTB 71768520 IC50 >= 10000 nM T11793 C4DS3F 2361 IC50 > 25000 nM T11793 C95JWC 68487 IC50 = 145000 nM T11793 CO0HB3 75473 Ki = 14000 nM T11793 CC0P7F 94378 IC50 = 6200 nM T11793 C6QB9N 126266 IC50 = 5100 nM T11793 CK8RD5 168114 IC50 = 8100 nM T11793 CJ34CF 168115 IC50 = 4300 nM T11793 C6LER8 210768 Ki = 1200 nM T11793 C6R5XN 595145 IC50 = 70800 nM T11793 CVRM18 595254 Ki = 30000 nM T11793 CTGL43 672443 IC50 = 50000 nM T11793 CGL5R1 683949 IC50 = 24000 nM T11793 C74MRA 702869 IC50 = 17700 nM T11793 C6DJ3Y 741004 IC50 = 3600 nM T11793 CSUL21 780263 IC50 = 50000 nM T11793 C06WCN 827839 IC50 = 9600 nM T11793 CZG18E 1201554 Ki = 43500 nM T11793 CRD18Y 2407524 IC50 = 70000 nM T11793 CQTY36 2650025 IC50 = 50000 nM T11793 CCQI26 3012527 IC50 = 50000 nM T11793 CAJQ53 3040177 Ki = 51500 nM T11793 C1ZC4D 4384047 IC50 = 50000 nM T11793 CZO2E5 4674678 IC50 = 50000 nM T11793 CBFV62 4817293 IC50 = 50000 nM T11793 CZM7D8 5281794 IC50 = 5800 nM T11793 CA5D1J 5289110 IC50 > 20000 nM T11793 CUL7A5 5471349 Ki = 5200 nM T11793 C48OIX 7074967 Ki = 71500 nM T11793 CA15IT 9796590 IC50 > 30000 nM T11793 CJDP76 9838675 EC50 = 600 nM T11793 C5LM9R 10221470 IC50 > 125000 nM T11793 CV5X8A 10224181 IC50 > 2500 nM T11793 C4A5SP 10379988 IC50 > 10000 nM T11793 CB0J3V 10383278 Ki = 5100 nM T11793 C8TPU0 10510985 Ki = 60000 nM T11793 CAC8P4 10647667 IC50 = 74300 nM T11793 CJPW17 10654534 Ki = 192000 nM T11793 CXK63D 10829689 IC50 = 44800 nM T11793 CZS9Q5 10899427 IC50 = 21600 nM T11793 C1A8HL 11171679 Ki > 400000 nM T11793 C1XR3I 11206290 Ki = 26100 nM T11793 CJ1O6V 11207072 IC50 = 5300 nM T11793 CMHY80 11229234 Ki = 179000 nM T11793 CF5YS9 11310529 Ki > 400000 nM T11793 CMQD35 11321674 Ki > 400000 nM T11793 CU72EY 11344157 Ki = 73000 nM T11793 C5FG8X 11355925 IC50 = 128000 nM T11793 C1BOK3 11378800 Ki = 3100 nM T11793 CZIC23 11389737 IC50 = 72100 nM T11793 CYL06Q 11389927 IC50 = 11800 nM T11793 CW57BU 11480732 IC50 = 83100 nM T11793 CB59HM 11570626 IC50 = 23000 nM T11793 CM7LS0 11612187 IC50 = 21000 nM T11793 CT4BE7 11641076 IC50 = 28000 nM T11793 C1T8XZ 11993865 Ki = 33700 nM T11793 CBZ83S 11993868 Ki = 5100 nM T11793 C7A1EZ 11993870 Ki = 33200 nM T11793 C4XP2N 11993872 Ki = 900 nM T11793 CWT0S3 11993875 Ki = 600 nM T11793 C7I9PF 13557523 Ki > 400000 nM T11793 C1G0EZ 13957609 IC50 = 8400 nM T11793 CT4RL1 15778480 IC50 = 217000 nM T11793 CDU1L0 16041411 IC50 > 60000 nM T11793 CJU50N 16072099 IC50 > 100000 nM T11793 CVJ4O1 16654686 Ki > 300000 nM T11793 C92NRU 16727109 IC50 > 40000 nM T11793 CW85LQ 16745311 IC50 = 100000 nM T11793 CKH72O 20115797 IC50 = 28800 nM T11793 CY9B5M 21257907 IC50 > 4000 nM T11793 CDL4G9 23645678 IC50 > 200000 nM T11793 CB4LY1 24857598 IC50 > 10000 nM T11793 CE95WV 24970356 IC50 = 5340 nM T11793 CXDF80 25034348 IC50 > 50000 nM T11793 C7EQ5T 25054288 IC50 > 10000 nM T11793 C6Z3CE 25057124 IC50 > 10000 nM T11793 CMH41V 25069448 IC50 = 11850 nM T11793 CBRM65 25074167 IC50 = 10400 nM T11793 C0XHA2 25180109 IC50 < 50000 nM T11793 C90UKD 25180304 IC50 = 47400 nM T11793 C6ZE9H 25180500 IC50 < 50000 nM T11793 C8CY6O 25205318 IC50 > 10000000 nM T11793 CY1M9Q 25205319 IC50 > 10000000 nM T11793 CC9S5U 28412206 IC50 < 100 nM T11793 C0FA2X 40680501 IC50 = 50000 nM T11793 C5E6UL 43388611 IC50 = 5500 nM T11793 C5L6WO 44194849 IC50 > 10000 nM T11793 C4W0SH 44247585 IC50 > 40000 nM T11793 CM6V4C 44388606 IC50 = 146000 nM T11793 CKV1H9 44388612 IC50 > 300000 nM T11793 CGU79D 44388657 IC50 = 256000 nM T11793 CAWL05 44428924 IC50 > 100000 nM T11793 CH54CO 44589824 IC50 = 19900 nM T11793 C89LHN 44589825 IC50 = 12600 nM T11793 C7UAT9 46174270 IC50 > 30000 nM T11793 C2M9XO 46835914 IC50 > 40000 nM T11793 C9CR0E 46835922 IC50 > 40000 nM T11793 CT6MJ2 46852951 IC50 > 50000 nM T11793 CO3P0J 46866604 IC50 > 30000 nM T11793 CJ3FM4 46925833 IC50 = 36160 nM T11793 CF14PE 46947264 IC50 > 30000 nM T11793 CX6NK2 47144386 IC50 = 9900 nM T11793 C3DN7U 49843520 IC50 > 10000 nM T11793 CECB91 49843530 IC50 > 31000 nM T11793 CF91RS 49843531 IC50 = 8150 nM T11793 CY46CB 49843532 IC50 > 50000 nM T11793 CMV6Y2 49868651 IC50 > 40000 nM T11793 CO0Y6K 49872677 IC50 > 10000 nM T11793 CJWE29 49872771 IC50 > 10000 nM T11793 CK9VE4 49872772 IC50 > 10000 nM T11793 CFP14Q 49872867 IC50 > 10000 nM T11793 C83CTW 49872868 IC50 > 10000 nM T11793 CLB34U 49872872 IC50 > 10000 nM T11793 CAM1D0 49873181 IC50 > 10000 nM T11793 CFT6V9 49873225 IC50 = 4900 nM T11793 C1N4YP 50908737 IC50 > 10000 nM T11793 CJD25G 52920263 IC50 = 16000 nM T11793 C1YLX8 52941699 IC50 > 10000 nM T11793 C34WMT 52942456 IC50 > 10000 nM T11793 C7SAC6 52948857 IC50 > 10000000 nM T11793 C0T5VA 53467975 IC50 > 11000 nM T11793 C2XHO3 53468206 IC50 > 11000 nM T11793 CUIB93 56679632 IC50 = 206000 nM T11793 CKY51C 56847605 IC50 = 54000 nM T11793 CZRQ14 56929159 IC50 = 54000 nM T11793 C90URY 56929249 IC50 = 54000 nM T11793 CWB5H7 56953768 IC50 = 10500 nM T11793 CS0HF1 56953769 IC50 = 15400 nM T11793 CPJ7X3 56953770 IC50 = 14800 nM T11793 CK7M6W 56953771 IC50 = 16600 nM T11793 CO96BR 56953896 IC50 = 50000 nM T11793 CJ0WM6 56953897 IC50 = 21400 nM T11793 C4UV1D 56953898 IC50 = 14400 nM T11793 CPKI96 56954010 IC50 = 4400 nM T11793 C6Q8BZ 56954011 IC50 = 1100 nM T11793 C5G4UX 56954012 IC50 = 15500 nM T11793 C8UQ2S 56954013 IC50 = 2000 nM T11793 CHQA53 56954137 IC50 = 50000 nM T11793 CZGE53 56954138 IC50 = 21800 nM T11793 C37SMZ 57505249 IC50 > 100000 nM T11793 C7I4QD 57519510 IC50 > 50000 nM T11793 C6JKM0 58834906 IC50 > 100000 nM T11793 CF9Z0L 58834953 IC50 > 26000 nM T11793 C4PWA9 58835024 IC50 > 40000 nM T11793 CCR4T7 58835217 IC50 > 73000 nM T11793 CFDG19 59401765 IC50 > 30000 nM T11793 CC5QW1 59401793 IC50 > 30000 nM T11793 CNOI48 59401886 IC50 > 30000 nM T11793 CTL97W 60151476 IC50 > 45000 nM T11793 C2D3HQ 60168069 IC50 > 200000 nM T11793 C1LB6D 66558197 IC50 = 4800 nM T11793 C7UKS4 66558379 IC50 > 100000 nM T11793 CCK6E5 66558639 IC50 = 75000 nM T11793 C40FKD 66898172 IC50 > 50000 nM T11793 C7TJ9X 66898814 IC50 > 50000 nM T11793 CFM6H7 67049587 IC50 > 100000 nM T11793 C4R8OG 67401728 IC50 > 30000 nM T11793 CHD80I 69937162 IC50 > 50000 nM T11793 CAR2N8 69937236 IC50 > 50000 nM T11793 CN7X0U 69937257 IC50 > 50000 nM T11793 C7VJ6A 70647728 IC50 > 40000 nM T11793 CUCQ24 70874317 IC50 > 100000 nM T11793 C8LCK6 70874412 IC50 = 4500 nM T11793 C1H7VK 70874453 IC50 = 10000 nM T11793 CJF91M 70874544 IC50 = 41000 nM T11793 C9EWB8 70874603 IC50 > 100000 nM T11793 C82PUD 70874605 IC50 = 39000 nM T11793 C8Q4LJ 70874786 IC50 = 50000 nM T11793 CF1G3K 70874916 IC50 > 100000 nM T11793 C30AJI 70914208 IC50 = 74000 nM T11793 C71AZM 70914219 IC50 = 56000 nM T11793 C2TC8W 70914230 IC50 = 51000 nM T11793 C8V5NF 70914234 IC50 = 43000 nM T11793 CP8HI7 70914358 IC50 > 100000 nM T11793 CS9OV5 71315139 IC50 = 88000 nM T11793 CC07KL 71662263 IC50 > 25000 nM T11793 CO1B9W 71662264 IC50 > 25000 nM T11793 CI0VR5 71662265 IC50 > 25000 nM T11793 CHW2T7 71662266 IC50 = 6290 nM T11793 CY9VC3 71662267 IC50 = 7120 nM T11793 C1MHC9 71662268 IC50 = 6620 nM T11793 CO57BK 71662269 IC50 > 25000 nM T11793 CZ01TB 71662427 IC50 > 25000 nM T11793 CHKX52 71662428 IC50 > 25000 nM T11793 C6PF9B 71662429 IC50 = 4080 nM T11793 C3DZ1E 71662430 IC50 > 25000 nM T11793 CPH76Z 71662431 IC50 > 25000 nM T11793 CKQ42X 71662432 IC50 > 25000 nM T11793 CXFB14 71662433 IC50 > 25000 nM T11793 CJHI28 71770158 IC50 > 20000 nM T11793 C9LU5Q 71770282 IC50 > 20000 nM T11793 C5JV1P 71812623 EC50 > 100000 nM T11793 CWT7K2 72205601 IC50 > 20000 nM T11793 C4G2UR 72695027 IC50 > 10000 nM T11793 CDFO42 72695136 IC50 > 10000 nM T11793 C3J0ZB 72725671 IC50 > 20000 nM T11793 C9WU2M 72950813 IC50 > 100000 nM T11793 CPG73S 73417116 IC50 = 6240 nM T11793 CWG4T2 78209992 IC50 > 50 nM T11793 CN9MO7 86271494 IC50 >= 19000 nM T11793 CKQ71X 86288935 IC50 = 33870 nM T11793 C5MR9K 89777151 EC50 > 50000 nM T11793 CE4IT5 90408860 IC50 >= 19000 nM T11793 CUQ1W0 91810395 IC50 > 50000 nM T11793 CWTO83 91810751 IC50 > 10000 nM T11793 CC9B6T 91820646 IC50 > 18000 nM T11793 CU1G3S 91933941 IC50 > 10000 nM T11793 CR4DE7 118175009 IC50 > 10000 nM T11793 C6HSC3 118217854 IC50 > 10000 nM T11793 CEKH57 118217858 IC50 > 10000 nM T11793 CB41MH 118560618 IC50 = 52000 nM T11793 C5BOQ1 118753201 Ki > 30000 nM T11793 C65ZYO 121332604 IC50 > 3000 nM T11793 C92NOH 121332654 IC50 > 3000 nM T11793 CNBH32 121332727 IC50 > 3000 nM T11793 C91PVZ 121428416 IC50 > 10000 nM T11793 C14FGL 122187534 IC50 > 20000 nM T11793 CB7IJ0 122188138 IC50 > 20000 nM T11793 CTI2V5 122192293 IC50 > 40000 nM T11793 C1C9LI 122246967 IC50 = 22000 nM T11793 C5ZY7L 124114343 IC50 > 50000 nM T11793 CDS92J 126483508 IC50 > 50000 nM T11793 CI3X9L 127049803 IC50 = 35670 nM T11793 C2O5LX 127049804 IC50 = 31760 nM T11793 C5OE2H 127053611 IC50 > 20000 nM T11793 CR8HP6 129281194 IC50 > 10000 nM T11793 CZ5H2B 132020452 IC50 = 9700 nM T11793 CP8A1Q 132020575 IC50 > 40000 nM T11793 CH8DP7 132220479 IC50 > 20000 nM T11793 CACJ46 132489333 IC50 > 25000 nM T11793 CS4BM3 135236903 IC50 > 50000 nM T11793 C7K4PA 135412054 IC50 > 20000 nM T11793 C31VAN 135412231 IC50 > 20000 nM T11793 C8R4FB 135546884 IC50 > 20000 nM T11793 CQ10OF 136240980 IC50 > 20000 nM T11793 C0PL4B 137434175 IC50 > 30000 nM T11793 C58ISN 137643139 IC50 = 10000 nM T11793 CLT73G 137647199 IC50 > 10000 nM T11793 C38FXZ 137653443 IC50 > 20000 nM T11793 C17LIA 137655641 IC50 > 33000 nM T11793 C96QPV 137662004 IC50 > 5000 nM T11793 C6KYD7 137700754 IC50 > 10000 nM T11793 CPTE92 138319693 IC50 > 10000 nM T11793 C1XSH7 138594194 IC50 > 10000 nM T11793 CGA12N 141473855 IC50 = 23570 nM T11793 C2YC6F 141473885 IC50 = 29380 nM T11793 C17XZS 142727681 IC50 > 25000 nM T11793 CXJ07F 145949470 IC50 = 4600 nM T11793 CI3V6Y 145950358 IC50 = 20000 nM T11793 CLZ54T 145950740 IC50 = 4100 nM T11793 C4FM3C 145951105 IC50 = 19000 nM T11793 CLV0G6 145951167 IC50 = 5800 nM T11793 CG5OW3 145951998 IC50 = 364000 nM T11793 C4LJV9 145952024 IC50 = 3500 nM T11793 C1QA6W 145952070 IC50 = 1300 nM T11793 CC7IP8 145952109 IC50 = 3500 nM T11793 C9D5MZ 145952745 IC50 = 11000 nM T11793 CRN85T 145952991 IC50 > 25000 nM T11793 CA7W2O 145953059 IC50 = 370 nM T11793 C5LB7M 145953999 IC50 = 7800 nM T11793 CN5L4K 145954640 IC50 = 230 nM T11793 CQ5SN1 145955289 IC50 = 73 nM T11793 C7N6CA 145956935 IC50 = 62 nM T11793 CBFU43 145957229 IC50 = 93 nM T11793 C20EDK 145957568 IC50 = 1200 nM T11793 C3B0YE 145957778 IC50 = 5000 nM T11793 CID3G5 145958087 IC50 = 13000 nM T11793 CM8U9A 145958674 IC50 = 120 nM T11793 CBF54O 145958967 IC50 = 3900 nM T11793 CB5XW7 145959080 IC50 = 180 nM T11793 CLS3W5 145959177 IC50 > 25000 nM T11793 CLJE41 145959897 IC50 > 25000 nM T11793 CW1GO5 145960043 IC50 = 3000 nM T11793 CDKY72 145960338 IC50 = 40000 nM T11793 CZ83QK 145960490 IC50 > 50000 nM T11793 CKLA91 145962920 IC50 = 87 nM T11793 CXF9E7 145972420 IC50 = 60 nM T11793 C56HYE 145974067 IC50 = 850 nM T11793 CJN96Q 145974556 IC50 = 13000 nM T11793 CWA6L3 145981037 IC50 = 12800 nM T11793 CMRQ02 145987862 IC50 > 20000 nM T11793 C7GK3H 145990715 IC50 = 84700 nM T11793 CE1L5T 145992719 IC50 > 20000 nM T11793 CMIH10 145993513 IC50 = 14900 nM T11793 CHJ79V 145997874 IC50 > 10000 nM T11793 C7F6SU 146047134 IC50 > 200000 nM T11793 C2J9YV 154727580 IC50 = 62000 nM T11793 CF2CU8 155510758 IC50 > 30000 nM T11793 CDV4Z6 155515709 IC50 = 258000 nM T11793 C28HEF 155519544 IC50 = 85400 nM T11793 C7SEX2 155529894 IC50 > 50000 nM T11793 CRY3A2 155548898 IC50 > 30000 nM T11793 C8Q2FG 155555556 IC50 > 20000 nM T11793 CKX10W 155562129 IC50 > 50000 nM T11793 CWOE21 155564042 IC50 > 30000 nM T11793 D00AWM 9826520 IC50 > 10000000 nM T11793 D00YNA 25093374 IC50 > 4000 nM T11793 D01ARE 44388719 IC50 = 6800 nM T11793 D01UYI 5281607 IC50 > 25000 nM T11793 D02EAP 11993867 Ki = 5300 nM T11793 D02GFK 25034431 IC50 > 50000 nM T11793 D03YHZ 25147692 IC50 = 100000 nM T11793 D06CWR 24754344 IC50 = 16540 nM T11793 D06HOI 44249821 IC50 > 40000 nM T11793 D06QFO 11332763 Ki = 95500 nM T11793 D06TRS 23646069 Ki = 1900 nM T11793 D07WLT 25180108 IC50 < 50000 nM T11793 D08IDC 24827305 IC50 > 25000 nM T11793 D09CPC 13728862 IC50 < 50000 nM T11793 D0A0GU 44247568 IC50 > 10000 nM T11793 D0G9WP 18407230 IC50 < 50000 nM T11793 D0I7GE 11790 IC50 = 13000 nM T11793 D0J1IE 11993873 Ki = 46900 nM T11793 D0K4LS 10691533 IC50 = 24800 nM T11793 D0M0IQ 11210706 IC50 = 9000 nM T11793 D0NM0P 25093389 IC50 > 4000 nM T11793 D0O1HH 11263510 Ki = 82500 nM T11793 D0P8PK 10192730 IC50 = 13400 nM T11793 D0Q5PC 6468 Ki = 10000 nM T11793 D0V2QH 24894072 IC50 = 7960 nM T11793 D0VD5O 11148236 Ki = 5900 nM T11793 D0Y1YR 442793 IC50 = 40800 nM T11793 D0YP4A 11993866 Ki = 1100 nM T11793 D0YQ8U 11993871 Ki = 3800 nM T36581 D0E3TC 44259 IC50 = 3550 nM T36581 D03BNU 59604787 IC50 > 10000 nM T36581 D0T3ME 156422 IC50 > 30000 nM T36581 CJWX69 3848929 IC50 > 200000 nM T36581 CBOP58 11293798 Ki > 10000 nM T36581 C26BZX 11362471 Ki > 10000 nM T36581 CWXB93 11397177 Ki > 10000 nM T36581 CJ9KN7 11683817 IC50 > 10000 nM T36581 C8E4TS 11992146 IC50 = 1100 nM T36581 C30UFT 16066811 IC50 = 4520 nM T36581 CUR7H3 16719862 IC50 = 660 nM T36581 CDMI50 23661564 IC50 = 90000 nM T36581 C9URB7 44441149 IC50 = 160000 nM T36581 C3VRO9 44557921 IC50 > 10000 nM T36581 CY3HW5 46224684 IC50 = 3800 nM T36581 CLS29B 46872626 IC50 > 10000 nM T36581 C2O8RZ 46886323 IC50 > 1000 nM T36581 C8ZRE3 53356518 IC50 = 213 nM T36581 C8NA4L 53384644 IC50 > 30000 nM T36581 C1MR8Q 60097495 IC50 > 1000 nM T36581 CV63UL 67240318 IC50 > 10000 nM T36581 CKT60L 71455860 Ki > 9200 nM T36581 CJ2T9E 76332983 IC50 > 10000 nM T36581 CUO0C5 132156633 IC50 > 10000 nM T36581 C2MD1Q 155513187 IC50 > 10000 nM T36581 D00ERW 44444843 Ki > 9234 nM T36581 D00TBD 10461815 IC50 > 10000 nM T36581 D03DZO 11715767 IC50 = 57700 nM T36581 D0EW9J 10389239 IC50 = 210 nM T07087 D0AF6O 71731823 IC50 = 14 nM T07087 D0OB0F 5328940 IC50 = 134 nM T07087 D01SJT 11713159 IC50 = 13 nM T07087 D0E3TC 44259 IC50 = 10.6 nM T07087 D03BNU 59604787 IC50 > 10000 nM T07087 D0T3ME 156422 IC50 = 400 nM T07087 C6D4GE 3134 Ki > 10000 nM T07087 CHGS79 3551941 Ki > 10000 nM T07087 C4ER2C 10000911 IC50 = 1200 nM T07087 C7FT8B 11502189 IC50 = 120 nM T07087 CACS26 11561968 Ki > 2000 nM T07087 CN50CR 11596788 IC50 = 210 nM T07087 C5NB3M 11598628 IC50 = 11 nM T07087 CU0E8O 11690457 Ki > 2000 nM T07087 C52GLP 11963310 IC50 = 120 nM T07087 C08NEU 15945881 IC50 = 414 nM T07087 CW0S4T 16118986 IC50 = 14 nM T07087 C21OUW 21952403 IC50 > 1100 nM T07087 C23ZPO 21952457 IC50 = 680 nM T07087 CS8D4H 21952489 IC50 = 190 nM T07087 C1TG0N 21952498 IC50 = 15 nM T07087 CLBP72 24798571 IC50 = 3184 nM T07087 C64KQP 25203958 IC50 = 637 nM T07087 CFMU29 25229638 IC50 = 50 nM T07087 CKN0O6 25920890 IC50 = 154 nM T07087 C3VRO9 44557921 IC50 > 10000 nM T07087 CUR98X 44562852 IC50 = 67 nM T07087 C0P2TQ 44562903 IC50 = 600 nM T07087 CF5Z1T 44562904 IC50 > 10000 nM T07087 CEJ8Y3 44562905 IC50 > 3000 nM T07087 CB8W7D 44562906 IC50 > 1000 nM T07087 CIQ36A 44562948 IC50 = 580 nM T07087 CBU64Q 44562949 IC50 = 1800 nM T07087 CF7I1N 44562995 IC50 = 17 nM T07087 C4EP1W 44562996 IC50 = 49 nM T07087 C2U3YS 44563035 IC50 = 53 nM T07087 CT03OG 44563036 IC50 = 33 nM T07087 CBWH32 44563037 IC50 = 5 nM T07087 CQC28T 44563059 IC50 = 143 nM T07087 CV3JH2 44563060 IC50 = 25 nM T07087 CZW0B1 44563061 IC50 = 95 nM T07087 C1Q7WR 44563062 IC50 = 35 nM T07087 CW0KF5 44563103 IC50 = 6 nM T07087 CSK2T1 44563136 IC50 = 2 nM T07087 C6QT0J 44622837 IC50 = 110 nM T07087 CP7L4W 45265983 IC50 = 31 nM T07087 CL1Z7W 45274615 IC50 = 170 nM T07087 C4AD7X 45274823 IC50 = 1500 nM T07087 CX5S8P 45274824 IC50 = 2800 nM T07087 C6C9WM 45274825 IC50 = 50 nM T07087 CMS63Y 45274934 IC50 = 44 nM T07087 CP5LH0 45274936 IC50 = 200 nM T07087 CAG3R0 45275054 IC50 = 430 nM T07087 CQU52A 45275055 IC50 = 53 nM T07087 CXZ2S5 45275165 IC50 = 33 nM T07087 CW08BK 45275166 IC50 = 1000 nM T07087 C43NVG 45275167 IC50 = 49 nM T07087 C8NA4L 53384644 IC50 > 30000 nM T07087 CWAY25 54586353 IC50 = 95 nM T07087 C8AB1J 54759606 Ki = 340 nM T07087 C1MR8Q 60097495 IC50 > 1000 nM T07087 CV63UL 67240318 IC50 > 10000 nM T07087 C3ETH7 70678491 IC50 = 1200 nM T07087 C7UYO2 70678492 IC50 = 78 nM T07087 CET75L 70692073 IC50 = 21 nM T07087 CC6OY7 71450691 IC50 = 25 nM T07087 CW1P5B 71450692 IC50 = 6.4 nM T07087 CN58DI 71450722 IC50 = 31 nM T07087 C5Z6EG 71452514 IC50 = 75 nM T07087 C76MBZ 71452515 IC50 > 100000 nM T07087 C0G8QT 71454271 IC50 = 57 nM T07087 CI03HX 71454272 IC50 = 3819 nM T07087 CMN73W 71454308 IC50 = 173 nM T07087 C0ML9S 71456031 IC50 = 12.5 nM T07087 CPEQ71 71456058 IC50 = 225 nM T07087 CT8UI0 71457834 IC50 = 398 nM T07087 CME4V0 71459744 IC50 = 1700 nM T07087 CTM3G8 71459745 IC50 = 361 nM T07087 C05XRA 71459746 IC50 = 1350 nM T07087 C5U6OG 71459747 IC50 = 429 nM T07087 CPDR94 71459748 IC50 = 69 nM T07087 C4V7QO 71461467 IC50 > 10000 nM T07087 CB3SO2 71567006 IC50 > 10000 nM T07087 CDJY72 71568837 IC50 = 6800 nM T07087 C8CAG7 71578921 IC50 > 30000 nM T07087 CL0T7B 76322219 IC50 = 10143 nM T07087 CMXH52 134130812 IC50 = 3.1 nM T07087 CMAJ86 134132390 IC50 = 3.5 nM T07087 CG9S2T 134132953 IC50 = 1.9 nM T07087 C3FXQ8 134133959 IC50 = 6625 nM T07087 CQ8SO0 134134585 IC50 = 1.5 nM T07087 CKGX09 134136179 IC50 = 122 nM T07087 CC82TI 134141407 IC50 = 201 nM T07087 C7QNE8 134143033 IC50 = 30 nM T07087 C5WE2S 134147409 IC50 = 0.67 nM T07087 CV02ZU 134149369 IC50 = 256 nM T07087 C6XHZ0 134149712 IC50 = 26 nM T07087 C04SWY 134150465 IC50 = 19.5 nM T07087 CZBC58 134153003 IC50 = 2.7 nM T07087 CJ47PZ 134153599 IC50 = 1.55 nM T07087 C73UZY 134155285 IC50 = 2.6 nM T07087 C1IQ6Y 134155909 IC50 = 0.9 nM T07087 CP9MH0 134156043 IC50 = 0.84 nM T07087 C2UJ9A 134156448 IC50 = 1.31 nM T07087 CU9R3M 136036273 Ki > 10000 nM T07087 C2VTB1 136216700 IC50 = 141 nM T07087 C2MD1Q 155513187 IC50 > 10000 nM T07087 D00SEC 3641059 Ki = 933.25 nM T07087 D02NNT 53232451 IC50 = 129 nM T07087 D02QAZ 11612883 IC50 > 1000 nM T07087 D0A0JL 2052 Ki = 162.18 nM T07087 D0AY0F 70698427 IC50 > 10000 nM T07087 D0E1QI 9549297 Ki = 10.47 nM T07087 D0K5UF 72710568 IC50 = 12 nM T07087 D0Y5RO 4566 Ki > 10000 nM T51282 D0B5LF 448042 Ki = 25.12 nM T51282 D00UET 15604510 IC50 = 186.21 nM T51282 D01NEC 51042438 IC50 = 125 nM T51282 D01ZAQ 25227436 IC50 = 470 nM T51282 D02NNV 3038525 IC50 > 5000 nM T51282 D02ZQS 16095342 IC50 = 1.8 nM T51282 D03KKR 3547 Ki = 100 nM T51282 D08HOM 46207586 IC50 = 456 nM T51282 D08ZPO 448043 IC50 = 5 nM T51282 D09XZL 56962369 IC50 = 2200 nM T51282 D0E3TC 44259 IC50 = 0.64 nM T51282 D0LL4Y 135564531 IC50 = 430 nM T51282 D0MS3Z 16725726 IC50 = 890 nM T51282 D0U5UC 11950170 Ki = 40 nM T51282 D0U9LT 9810884 IC50 = 120 nM T51282 D03BNU 59604787 IC50 > 10000 nM T51282 D00YYO 118888942 IC50 = 110 nM T51282 D05PTF 118888905 IC50 = 1900 nM T51282 D0CW9Q 56596554 IC50 = 650 nM T51282 D0U5IW 118888913 IC50 = 450 nM T51282 D0YD7S 118888923 IC50 = 84 nM T51282 D0T3ME 156422 IC50 > 30000 nM T51282 CWT4N9 4216 IC50 = 38000 nM T51282 C8BZK3 5711 IC50 = 200 nM T51282 CWI59L 88012 IC50 = 181300 nM T51282 CHAL37 482056 IC50 = 480 nM T51282 CP9AM1 599038 Ki = 330 nM T51282 CE2G1Z 607858 Ki = 360 nM T51282 CN8SU3 684961 Ki = 1900 nM T51282 C5LHO7 753058 Ki > 3300 nM T51282 CSE25J 2123970 Ki = 540 nM T51282 C49YTC 2227730 IC50 = 270000 nM T51282 CF49GB 2824220 IC50 = 1500 nM T51282 CIU9K1 3049109 IC50 = 75500 nM T51282 CZX36A 4421488 IC50 = 157100 nM T51282 C5O3TE 4801910 Ki > 2500 nM T51282 CI4DE0 4803142 Ki = 83 nM T51282 C6AD8F 5038004 Ki = 930 nM T51282 CEU1N6 5056270 IC50 = 13 nM T51282 CHQ7M1 8123789 Ki = 120 nM T51282 CQV9N0 8123825 Ki = 130 nM T51282 C4KEJ2 9860439 IC50 = 570 nM T51282 CV50OB 9863672 IC50 = 51 nM T51282 CE40AW 9885023 IC50 = 30 nM T51282 C9O3XQ 9901617 IC50 = 46 nM T51282 CF9A5O 10125353 Ki = 660 nM T51282 CM79VS 10149184 Ki = 450 nM T51282 C69DHW 10158652 IC50 < 16000 nM T51282 CC8XJ5 10171595 Ki = 590 nM T51282 CB28QI 10171783 Ki = 810 nM T51282 CL7FI4 10171832 Ki > 5000 nM T51282 CJ39UQ 10236371 Ki = 720 nM T51282 C7SFI1 10296883 IC50 > 10000 nM T51282 C87AML 10402473 Ki = 1100 nM T51282 CLZK93 11189172 IC50 = 5 nM T51282 CR6U2M 11196984 IC50 = 550 nM T51282 CM6DO0 11233873 IC50 = 14 nM T51282 C0OZW2 11247002 IC50 = 8 nM T51282 C49NET 11256399 IC50 = 3 nM T51282 CN16LZ 11269477 IC50 = 9 nM T51282 CBOP58 11293798 Ki > 10000 nM T51282 CA63NG 11339681 IC50 = 4 nM T51282 COW1S8 11360518 IC50 = 51 nM T51282 C26BZX 11362471 Ki > 10000 nM T51282 C9UI3O 11373846 IC50 = 14 nM T51282 CWXB93 11397177 Ki > 10000 nM T51282 CHOV59 11404963 IC50 = 18 nM T51282 CONW29 11453116 IC50 = 9 nM T51282 CS2YO1 11492918 Ki > 3300 nM T51282 C17UMV 11495551 IC50 = 5200 nM T51282 CEK1G9 11503627 IC50 = 68000 nM T51282 CNSX26 11515518 Ki = 5 nM T51282 C3VXY4 11518055 IC50 > 10000 nM T51282 CT1WQ3 11525337 Ki = 3 nM T51282 CGC86O 11525338 Ki = 6 nM T51282 CY5F0M 11526080 IC50 = 288 nM T51282 CE9R7D 11530100 IC50 = 120000 nM T51282 CIN49V 11531981 IC50 = 180 nM T51282 C9HSI4 11531982 IC50 = 8 nM T51282 CXL01N 11536733 IC50 = 25000 nM T51282 CR92GA 11537005 IC50 = 160 nM T51282 CTG83F 11539329 Ki > 9100 nM T51282 C5T0GN 11545280 IC50 = 863 nM T51282 C82BTJ 11547150 Ki = 8 nM T51282 C7IOJ0 11548023 IC50 = 6 nM T51282 CME81U 11560302 IC50 = 2300 nM T51282 C17MUY 11561279 Ki = 19 nM T51282 CN08CJ 11561907 IC50 = 250 nM T51282 CACS26 11561968 Ki < 5 nM T51282 CC84NJ 11569498 IC50 = 75 nM T51282 C4AL8Z 11575817 IC50 = 2500 nM T51282 CSW50Y 11581362 Ki = 3 nM T51282 CMIL86 11590363 Ki > 9100 nM T51282 CHI4R8 11590594 IC50 = 46 nM T51282 CUGJ03 11590642 IC50 = 104 nM T51282 C0TA5Q 11597345 IC50 = 129 nM T51282 C1ZUJ6 11604313 IC50 = 105 nM T51282 CYEN01 11605242 Ki = 2 nM T51282 C39KYQ 11605996 IC50 = 150 nM T51282 CJ5K9X 11609495 IC50 = 1500 nM T51282 C5XC9Q 11611566 IC50 > 10000 nM T51282 C71WAD 11615485 Ki > 3300 nM T51282 CP2MJ8 11620539 IC50 = 68 nM T51282 CQ2ZX6 11632274 Ki = 6 nM T51282 C3NDK9 11633229 IC50 = 1290 nM T51282 C8C3PR 11639062 Ki = 14 nM T51282 C9T6SC 11640926 Ki > 9100 nM T51282 CJS28X 11641672 IC50 = 5 nM T51282 CQRB62 11641686 IC50 = 3 nM T51282 CM08LS 11648365 IC50 > 10000 nM T51282 CJ4Z7K 11649154 IC50 = 15 nM T51282 CM2T8F 11656187 IC50 = 4 nM T51282 C3E0TV 11663187 IC50 = 2 nM T51282 CQGI52 11667631 IC50 = 9600 nM T51282 CU0E8O 11690457 Ki = 2 nM T51282 C25STN 11690618 IC50 > 10000 nM T51282 C3YKD0 11691434 Ki = 10 nM T51282 C65FVB 11694317 Ki > 3300 nM T51282 CXS4V3 11694866 IC50 = 4600 nM T51282 COH3C4 11697546 IC50 = 105 nM T51282 C43TXY 11703935 IC50 > 10000 nM T51282 CB0AP2 11705863 Ki < 1 nM T51282 C70LWD 11712638 Ki = 3 nM T51282 C6AH2S 11716019 IC50 = 37000 nM T51282 CJM6I4 11717275 Ki = 3 nM T51282 C5ISQ9 11751266 IC50 = 8 nM T51282 CJS3M6 11772907 IC50 = 13 nM T51282 C3YRU7 15295578 IC50 = 60 nM T51282 CFPW41 16007116 Ki > 9100 nM T51282 C7Z4LV 16095343 IC50 = 5.6 nM T51282 CBG93R 16099843 IC50 = 30 nM T51282 C7OP3Q 16099844 IC50 = 1.8 nM T51282 CM4G5H 16099846 IC50 <= 1 nM T51282 CTN6O2 16099847 IC50 <= 1 nM T51282 CUJ09Z 16099848 IC50 <= 1 nM T51282 C97BRU 16099849 IC50 = 33 nM T51282 CNAH98 16099857 IC50 = 4.4 nM T51282 C6Y5GI 16099858 IC50 = 90 nM T51282 CN52XM 16099859 IC50 = 2 nM T51282 CI5AH6 16099860 IC50 <= 1 nM T51282 CZD9H6 16099861 IC50 <= 1 nM T51282 CQK6C4 16099866 IC50 = 2500 nM T51282 CZF23I 16124479 Ki = 2.512 nM T51282 C5VPH9 16129448 IC50 = 413 nM T51282 C94CRM 16222264 IC50 = 47.86 nM T51282 CML35S 16222265 IC50 = 331.13 nM T51282 CILJ71 16222356 IC50 = 239.88 nM T51282 CS8W9L 16222361 IC50 = 239.88 nM T51282 C4FO0C 16222562 IC50 = 524.81 nM T51282 CVZO20 16222567 IC50 = 588.84 nM T51282 CA20NM 16222570 Ki = 37.15 nM T51282 C1EDJ3 16222668 IC50 = 676.08 nM T51282 CUD0T7 16222673 IC50 = 870.96 nM T51282 CC9RM5 16344190 Ki = 170 nM T51282 C5XFD3 17757326 Ki = 120 nM T51282 CZT35Q 17838190 IC50 = 13900 nM T51282 CV78RB 18581471 Ki = 81 nM T51282 C4NWS6 22169775 IC50 = 7762.47 nM T51282 CW6OB1 23627212 IC50 > 9000 nM T51282 CG3VB6 23646578 IC50 < 10 nM T51282 CMD65I 23648890 IC50 = 19.95 nM T51282 CA12HF 24740244 IC50 = 230 nM T51282 CK60ZM 24758992 IC50 = 19 nM T51282 C7YG1N 24759534 IC50 = 360 nM T51282 C2UOE0 24766030 IC50 > 50000 nM T51282 CZY46J 24782989 IC50 = 165.96 nM T51282 C14WAZ 24782990 IC50 = 229.09 nM T51282 CPU52W 24783245 IC50 = 81.28 nM T51282 CLBP72 24798571 IC50 > 10000 nM T51282 CCP2M3 24822704 IC50 > 50000 nM T51282 CM28WD 24825721 IC50 > 10000 nM T51282 CZI9P0 24829572 Ki = 770 nM T51282 C4T3UC 24829746 Ki = 210 nM T51282 C47LFZ 24830567 Ki = 18 nM T51282 C9E7AU 24830568 Ki = 44 nM T51282 CJ4K3P 24830569 Ki = 45 nM T51282 CKL92Z 24830570 Ki = 22 nM T51282 C2K1OE 24830571 Ki = 10 nM T51282 CP4KZ1 24830882 Ki = 30 nM T51282 C4J6AD 24831672 Ki > 2500 nM T51282 C82YBD 24831841 Ki > 2500 nM T51282 CTXJ06 24832008 Ki = 110 nM T51282 C75KOR 24832012 Ki = 165 nM T51282 CZ2PQ6 24863113 IC50 = 14 nM T51282 CBYM61 24863535 IC50 = 180 nM T51282 C2S6QP 24877013 IC50 = 20 nM T51282 C9G5UN 24877483 IC50 = 360 nM T51282 C2PB0C 24877599 IC50 = 4200 nM T51282 C9LFA0 24877716 EC50 = 900 nM T51282 CA4N7R 24878052 IC50 = 28000 nM T51282 CKX4J8 24878054 IC50 > 10000 nM T51282 C0OBT6 24878164 IC50 = 8300 nM T51282 C78TNQ 24878165 IC50 = 13000 nM T51282 CR52WM 24878170 IC50 = 2900 nM T51282 CCBH01 24878396 IC50 = 580 nM T51282 CGQ62D 24878397 IC50 = 7200 nM T51282 C28FIM 24878398 IC50 = 20 nM T51282 CSE5Z1 24878503 EC50 = 3600 nM T51282 C1OHB3 24878504 IC50 = 2200 nM T51282 CK6I0C 24878508 IC50 = 9700 nM T51282 C9OMP1 24878615 IC50 = 8600 nM T51282 CC2M0I 24878617 IC50 = 60 nM T51282 C50EIA 24878618 EC50 > 10000 nM T51282 CWE0L7 24983829 IC50 = 316.23 nM T51282 C8O0JE 24985283 IC50 = 10000 nM T51282 CS3Q8B 24995659 Ki > 4000 nM T51282 C1ONA4 24996161 IC50 = 21 nM T51282 CA9F3Y 25023714 IC50 = 8 nM T51282 C8Z4PI 25023715 IC50 = 5 nM T51282 CV96QX 25023716 IC50 = 5 nM T51282 C5INV4 25023717 IC50 = 20 nM T51282 CPOH02 25023718 IC50 = 40 nM T51282 CW2MV8 25023720 IC50 = 158 nM T51282 CPB4S2 25023721 IC50 = 562 nM T51282 C8UL4O 25023722 IC50 = 126 nM T51282 CZ05HU 25023723 IC50 = 224 nM T51282 CSM1R7 25023724 IC50 = 1995 nM T51282 C4DF8X 25023725 IC50 = 501 nM T51282 CXFQ18 25023726 IC50 = 20 nM T51282 C13MHS 25023727 IC50 = 126 nM T51282 C1JEU6 25023729 IC50 = 500 nM T51282 C14NAT 25023731 IC50 = 500 nM T51282 C81XKW 25023732 IC50 = 1260 nM T51282 CFH80B 25023733 IC50 = 790 nM T51282 CR8JP7 25023735 IC50 = 890 nM T51282 C4W7LY 25023736 IC50 = 3980 nM T51282 CA6QU5 25023737 IC50 = 250 nM T51282 CX1HL8 25032704 Ki > 9110 nM T51282 CIH3E5 25093235 IC50 = 56 nM T51282 C0Q3WY 25093238 IC50 = 101 nM T51282 C8NU5G 25093239 IC50 = 129 nM T51282 CRX1C6 25093240 IC50 = 26 nM T51282 C1AGW7 25093241 IC50 = 6 nM T51282 CE50OH 25093242 IC50 = 11 nM T51282 CL9ZK6 25093243 IC50 = 10 nM T51282 C7BAN0 25262260 IC50 = 3.4 nM T51282 C0K2NM 41107723 Ki = 100 nM T51282 CWS37O 42618140 IC50 = 1258.93 nM T51282 C2JV3O 42618143 IC50 = 199.53 nM T51282 CG01BO 42618144 IC50 = 794.33 nM T51282 CO4FV0 42630578 IC50 > 10000 nM T51282 CO42DC 44138048 IC50 > 10000 nM T51282 CL65QV 44138049 IC50 > 10000 nM T51282 CLW80F 44160269 IC50 > 50000 nM T51282 CR7TY6 44197572 IC50 = 48 nM T51282 C1G2ZQ 44198874 IC50 = 33 nM T51282 CK73NR 44219749 IC50 > 50000 nM T51282 C23UAJ 44481840 IC50 > 2800 nM T51282 C4WRN5 44541014 IC50 = 50000 nM T51282 CRZ79W 44542926 IC50 = 310 nM T51282 CE0O4B 44543079 IC50 = 51 nM T51282 CQT48I 44543080 IC50 = 490 nM T51282 CCL85F 44575073 IC50 > 50000 nM T51282 CJX06P 44575126 IC50 > 50000 nM T51282 CE8FC7 44575127 IC50 > 50000 nM T51282 COY57J 44592504 IC50 = 2 nM T51282 C28QLM 44605035 IC50 > 50000 nM T51282 C75XHS 44605037 IC50 > 50000 nM T51282 CDN3C4 44622839 Ki = 2200 nM T51282 C5G0UA 44622840 Ki = 85 nM T51282 CG6UW5 44634494 IC50 = 3.5 nM T51282 CJ0F5Q 44819015 IC50 = 4300 nM T51282 CM3GX4 45102613 IC50 = 2390 nM T51282 CA4XQ3 45375859 IC50 = 2 nM T51282 CC95PQ 45375865 IC50 > 50000 nM T51282 CEOQ27 45375866 IC50 > 50000 nM T51282 C0FM5X 45381385 IC50 = 5536 nM T51282 CH0PJ3 45483176 IC50 = 400 nM T51282 CG8ER3 45483177 IC50 = 23 nM T51282 CUF6J2 45483178 IC50 = 2 nM T51282 C1FKP3 45483179 IC50 = 14 nM T51282 CALU07 45483184 IC50 = 1200 nM T51282 CBGO40 45483209 IC50 = 185 nM T51282 C2EO0W 45483210 IC50 = 57 nM T51282 C26GUE 45483248 IC50 = 8400 nM T51282 C30NRT 45483249 IC50 = 1000 nM T51282 C36YVC 45483250 IC50 = 7400 nM T51282 CQY54A 45483257 IC50 = 8300 nM T51282 CPF9I6 45483258 IC50 = 305 nM T51282 C37WKR 45483267 IC50 = 11 nM T51282 CWHI97 45483283 IC50 = 6 nM T51282 CGR94B 45483284 IC50 = 81 nM T51282 CW28FX 45483285 IC50 = 26 nM T51282 CV8H7Y 45483302 IC50 = 890 nM T51282 CR72XS 45483303 IC50 = 135 nM T51282 CU6W3S 45483304 IC50 = 118 nM T51282 CB70SK 45483322 IC50 = 87 nM T51282 CB76GJ 45483326 IC50 = 326 nM T51282 C5S8MA 45485083 IC50 > 8000 nM T51282 CW42YX 45487634 IC50 > 5000 nM T51282 C93OTW 46182713 IC50 = 10 nM T51282 C1MB8Y 46183900 IC50 = 1.2 nM T51282 C8ADR2 46214481 IC50 > 10000 nM T51282 CH0ZR1 46214482 IC50 = 3981.07 nM T51282 C2EZU8 46214649 IC50 = 6309.57 nM T51282 C5L1KH 46214650 IC50 > 10000 nM T51282 CRI6G5 46214652 IC50 > 10000 nM T51282 CRT51W 46214653 IC50 > 10000 nM T51282 CVW21C 46215644 IC50 = 2511.89 nM T51282 CZ58FY 46215814 IC50 = 1584.89 nM T51282 CO9H1K 46215816 IC50 = 3162.28 nM T51282 CT8G2A 46215988 IC50 = 15848.93 nM T51282 C28SJK 46215992 IC50 > 10000 nM T51282 C9JNT0 46216155 IC50 = 158.49 nM T51282 CD96WF 46216494 IC50 = 5011.87 nM T51282 C9LU8O 46216813 IC50 = 300 nM T51282 CY3HW5 46224684 IC50 = 400 nM T51282 CGA0E5 46226413 IC50 = 6000 nM T51282 CLW06M 46226414 IC50 > 10000 nM T51282 CI90DE 46226435 IC50 > 10000 nM T51282 C9XUZ7 46229921 IC50 = 4600 nM T51282 C05RZO 46229922 IC50 > 100000 nM T51282 CZ20AP 46230023 IC50 = 6900 nM T51282 CG3Y2V 46230024 IC50 = 6500 nM T51282 CF7J5W 46230025 IC50 = 2600 nM T51282 CRK5G7 46230026 IC50 = 42000 nM T51282 CO2SM4 46230027 IC50 = 10000 nM T51282 CG0T3I 46230078 IC50 = 48000 nM T51282 C6BVX1 46230079 IC50 = 6000 nM T51282 C1W7IZ 46230080 IC50 = 18000 nM T51282 C1SVR9 46230081 IC50 = 320 nM T51282 CI5CP4 46230131 IC50 = 610 nM T51282 CAI1J3 46230132 IC50 = 290 nM T51282 CJH61I 46230133 IC50 = 1800 nM T51282 C9N5GS 46230134 IC50 = 130 nM T51282 CC09NO 46230135 IC50 = 150 nM T51282 COQ5I4 46230172 IC50 = 170 nM T51282 CEF6C8 46230173 IC50 = 34 nM T51282 CVZ2F7 46230174 IC50 = 300 nM T51282 CDZ1V3 46230175 IC50 = 1400 nM T51282 CO3P0J 46866604 IC50 < 50000 nM T51282 CROT59 46871772 IC50 = 22 nM T51282 CLS29B 46872626 IC50 > 10000 nM T51282 CQIC19 46879806 IC50 = 180 nM T51282 CJOM49 46880136 IC50 = 17600 nM T51282 CNTS27 46883044 Ki = 180 nM T51282 C0DB5Z 46883045 Ki = 340 nM T51282 C9WE4S 46883122 Ki > 2500 nM T51282 CNTS75 46883123 Ki > 2500 nM T51282 CJS68B 46883124 Ki = 1300 nM T51282 CU3O2G 46883125 Ki = 2100 nM T51282 CH9RV4 46883165 Ki = 940 nM T51282 CT1K6A 46883166 Ki > 3300 nM T51282 CGZ1S4 46883167 Ki > 3300 nM T51282 C2VGJ9 46883168 Ki > 3300 nM T51282 CT5V8K 46883169 Ki > 3300 nM T51282 CRE96X 46885625 IC50 = 398 nM T51282 C2O8RZ 46886323 IC50 > 1000 nM T51282 CB28LG 46889347 EC50 = 2600 nM T51282 CLDJ97 46889348 IC50 = 30 nM T51282 CL1M9K 46889386 EC50 = 1900 nM T51282 CRS79N 46889387 EC50 = 1400 nM T51282 C4KS0X 46889388 IC50 = 400 nM T51282 CVOJ40 46889389 IC50 = 140 nM T51282 C6KVJ7 46889390 IC50 = 20 nM T51282 C2STG3 46889405 IC50 = 60 nM T51282 CDLP60 46889406 IC50 = 30 nM T51282 COJ7K0 46889855 IC50 = 1200 nM T51282 C3FIS5 46889888 IC50 > 100000 nM T51282 C3SBX1 46889889 IC50 = 7100 nM T51282 CXUO70 46890036 IC50 = 59 nM T51282 CZ2V8R 46890138 IC50 = 53 nM T51282 CA2Y8J 46901260 IC50 = 16 nM T51282 CSV5B9 46901859 IC50 = 30 nM T51282 CCL6T7 49870878 Ki = 34.67 nM T51282 CRCT70 50909914 IC50 = 794.33 nM T51282 C0XDI4 50909915 IC50 = 199.53 nM T51282 CUJL92 50909916 IC50 > 10000 nM T51282 C51DKX 50909917 IC50 > 10000 nM T51282 CUN2I8 50942209 IC50 = 4265.8 nM T51282 CM9KE0 50942210 IC50 = 3630.78 nM T51282 CX6PZ9 51003130 IC50 = 1 nM T51282 CYD4A2 51354035 IC50 = 3162.28 nM T51282 CW2T3N 51354036 IC50 > 10000 nM T51282 CH8NX6 51354037 IC50 > 10000 nM T51282 CK63DI 51354327 IC50 > 10000 nM T51282 CC6PZ4 51354328 IC50 > 10000 nM T51282 C2FVX4 51354329 IC50 > 10000 nM T51282 CV06QD 51354330 IC50 > 10000 nM T51282 CR3AC1 51354331 IC50 > 10000 nM T51282 CUXD62 51354613 IC50 > 10000 nM T51282 C3G1VK 51354899 IC50 = 15848.93 nM T51282 CK7NP1 51354900 IC50 > 10000 nM T51282 CEDN75 51354901 IC50 = 3162.28 nM T51282 CB0EU1 51355190 IC50 = 3162.28 nM T51282 CYZ03E 51356852 IC50 > 10000 nM T51282 CL3S8F 51356853 IC50 = 7943.28 nM T51282 C67DUF 51356854 IC50 > 10000 nM T51282 CAU2F6 51356855 IC50 > 10000 nM T51282 CD07RV 51356856 IC50 > 10000 nM T51282 CFM5I7 51357137 IC50 = 15848.93 nM T51282 CP6R5J 51357138 IC50 > 10000 nM T51282 CWCJ29 51357417 IC50 = 1995.26 nM T51282 CS9WE1 51357418 IC50 = 5011.87 nM T51282 C5G7BY 51357419 IC50 > 10000 nM T51282 CBM4P9 51357696 IC50 > 10000 nM T51282 C65MXB 51357954 IC50 = 630.96 nM T51282 CC41YU 52933429 IC50 = 8 nM T51282 COGV85 52933915 IC50 = 62 nM T51282 CB24WM 52933916 IC50 = 6 nM T51282 CEW2N3 52933917 IC50 = 40 nM T51282 C4D6ZP 52934146 IC50 = 21 nM T51282 CY8B9U 52934379 IC50 = 2 nM T51282 CD2S0G 52934380 IC50 > 20000 nM T51282 C2Q3AE 52934381 IC50 = 33 nM T51282 C6OA7K 52934832 IC50 = 480 nM T51282 CRDM19 52934834 IC50 = 6900 nM T51282 CU6W0S 52935059 IC50 = 13 nM T51282 CN5Y4M 52935061 IC50 = 1900 nM T51282 C5C2HR 52935064 IC50 = 500 nM T51282 C2BTX1 52935500 IC50 = 19 nM T51282 C5UOY3 52935712 IC50 = 88 nM T51282 CF54OU 52935714 IC50 = 710 nM T51282 CAN96R 52935715 IC50 < 1 nM T51282 C9OW2P 52935716 IC50 = 11 nM T51282 C0QF2H 52935717 IC50 = 110 nM T51282 C8IXZ0 52935926 IC50 = 5 nM T51282 C6SW7E 52936149 IC50 = 19 nM T51282 CWV3F9 52936150 IC50 = 720 nM T51282 C9JFX1 53316641 IC50 = 31.62 nM T51282 C5GQA6 53319060 IC50 > 100000 nM T51282 COR1L2 53319319 IC50 = 1949.84 nM T51282 C8XM9S 53319399 IC50 = 1479.11 nM T51282 CN5AS6 53319400 IC50 = 1698.24 nM T51282 CRI2V5 53320582 IC50 = 169.82 nM T51282 C97YXF 53320583 IC50 = 72.44 nM T51282 C8X1MP 53320584 IC50 = 57.54 nM T51282 C3UA4Y 53320702 IC50 = 588.84 nM T51282 CZ8IQ2 53320703 IC50 = 776.25 nM T51282 C3QP4L 53321582 IC50 = 575.44 nM T51282 CRY96M 53321650 Ki = 63.1 nM T51282 CJT1Q7 53321876 IC50 = 1778.28 nM T51282 C60OVM 53321877 IC50 = 120.23 nM T51282 CRN08I 53321993 IC50 = 1862.09 nM T51282 C3TUC4 53322817 IC50 = 6760.83 nM T51282 C9FC2P 53323357 IC50 = 1000 nM T51282 CRLD25 53325449 IC50 = 812.83 nM T51282 CR8UT4 53325978 IC50 = 426.58 nM T51282 C05DZE 53325979 IC50 = 3467.37 nM T51282 C0SWH5 53348216 IC50 > 40000 nM T51282 C8NA4L 53384644 IC50 > 30000 nM T51282 CNOA83 53492329 IC50 = 170 nM T51282 C8WFA5 53492330 IC50 = 27 nM T51282 CRN28X 54581311 IC50 > 10000 nM T51282 CUJM81 54765020 IC50 = 34 nM T51282 CQ28VE 54765021 IC50 = 89 nM T51282 CE0Y9O 54765203 IC50 = 12 nM T51282 C9V7LP 54765280 IC50 = 6 nM T51282 CG7F2E 56603818 IC50 = 30 nM T51282 CPC5D2 56603995 IC50 = 2510 nM T51282 CEBQ15 56604005 IC50 = 200 nM T51282 CFP56A 56604013 IC50 = 1000 nM T51282 CN9QD7 56643097 IC50 > 10000 nM T51282 C04QGT 57390719 IC50 = 1100 nM T51282 C2UZC6 57392519 IC50 = 19 nM T51282 CJ7HZ1 57392522 IC50 = 18 nM T51282 CJ1EI5 57392627 IC50 = 1100 nM T51282 C5RTO0 57394242 IC50 = 243 nM T51282 CJED53 57394243 IC50 = 121 nM T51282 CV4PQ1 57394244 IC50 = 1900 nM T51282 C4QK5J 57394245 IC50 = 240 nM T51282 C2OD1C 57394246 IC50 = 560 nM T51282 CAV49N 57394247 IC50 = 76 nM T51282 C5GYP7 57394348 IC50 = 870 nM T51282 CB6U0W 57395100 IC50 = 11 nM T51282 CYU92T 57395101 IC50 < 1 nM T51282 C8BKO6 57395998 IC50 = 23 nM T51282 C3WBE7 57395999 IC50 = 34 nM T51282 C70JBE 57396000 IC50 = 2 nM T51282 C6C7EN 57396001 IC50 = 500 nM T51282 CNH69U 57396872 IC50 = 76 nM T51282 CX24JF 57397800 IC50 = 280 nM T51282 C8R7HP 57397801 IC50 = 27 nM T51282 CBG3T9 57397802 IC50 = 1340 nM T51282 C07YVE 57397803 IC50 = 130 nM T51282 CWG07J 57399140 IC50 < 10 nM T51282 CV6X1C 57399460 IC50 = 37 nM T51282 CH84ZK 57399461 IC50 = 46 nM T51282 C3DR4A 57399462 IC50 = 6600 nM T51282 CG1FJ4 57399463 IC50 = 1000 nM T51282 CRA61Q 57399464 IC50 = 760 nM T51282 C6UGL7 57399465 IC50 = 170 nM T51282 C7DT8V 57400298 IC50 = 3 nM T51282 C0JAL7 57400299 IC50 = 30 nM T51282 CETA86 57401229 IC50 = 88 nM T51282 CHXD31 57401230 IC50 < 1 nM T51282 CT9NR3 57402100 IC50 = 3 nM T51282 CYUQ67 57402101 IC50 = 9 nM T51282 CL1WN9 57402102 IC50 = 8900 nM T51282 CC41DN 57402103 IC50 = 260 nM T51282 CSEA21 57402104 IC50 = 91 nM T51282 C1F3AS 57402971 IC50 = 48 nM T51282 C8XM3C 57403071 IC50 = 2100 nM T51282 CH5Q0E 57403072 IC50 = 1200 nM T51282 CN9G2Z 57403855 IC50 = 39 nM T51282 CI1A8M 57404048 IC50 = 1283 nM T51282 C8JQT0 57633016 Ki = 2 nM T51282 CKH8C1 57633047 Ki = 11 nM T51282 CSV52O 57633056 Ki = 2 nM T51282 CV6J8N 57633096 Ki < 1 nM T51282 C25KIP 57633210 Ki = 2 nM T51282 C2MD4C 57663921 IC50 = 9070 nM T51282 C8X6PU 57663989 IC50 = 1410 nM T51282 C6YAG9 57664030 IC50 = 1150 nM T51282 C9PKH2 57920206 IC50 = 514 nM T51282 C3V6MX 57920210 IC50 = 139 nM T51282 CBRV34 58310563 IC50 = 170 nM T51282 C81JXL 58310602 IC50 = 16.3 nM T51282 CBGN56 58310712 IC50 = 104 nM T51282 C2NV3R 59198239 IC50 = 30 nM T51282 CT3EW2 59292007 IC50 = 190 nM T51282 CXJ63M 59603829 IC50 = 780 nM T51282 CQEU96 59603842 IC50 = 17 nM T51282 CE37AG 60097359 Ki = 120 nM T51282 CGUC54 60097393 Ki = 220 nM T51282 C5MDR3 60097396 Ki = 140 nM T51282 CGI82D 60097406 Ki = 28 nM T51282 COH62U 60097413 IC50 = 7 nM T51282 CFMP63 60097457 Ki = 240 nM T51282 CPO71M 60097461 Ki = 47 nM T51282 CVD9Y1 60097467 Ki = 430 nM T51282 CJ5V4X 60097469 Ki = 10 nM T51282 CYC65S 60097478 Ki = 2500 nM T51282 C1MR8Q 60097495 IC50 = 8 nM T51282 CZT2A8 60097525 Ki = 510 nM T51282 C7DP4E 60097576 Ki = 350 nM T51282 CMF42W 60097605 Ki = 10 nM T51282 C31NRA 60097624 Ki = 88 nM T51282 CP5B0G 60097630 Ki = 26 nM T51282 C8LYG4 60097631 Ki = 45 nM T51282 CW1AE2 60097642 Ki = 17 nM T51282 CO27YK 60097661 Ki = 900 nM T51282 C2C3DJ 60097665 Ki = 61 nM T51282 C02BUA 60097693 Ki > 2500 nM T51282 C96PLJ 60097708 Ki = 70 nM T51282 C2VG1E 60097724 Ki = 530 nM T51282 CS73TH 60097732 Ki = 490 nM T51282 CK6WO0 66552478 IC50 < 10000 nM T51282 CNT5Z9 66743321 IC50 = 54 nM T51282 CM7O8P 66743326 IC50 = 44 nM T51282 CQ8PY7 66743332 IC50 = 130 nM T51282 CGD2H4 66743358 IC50 = 130 nM T51282 C6RX7H 66743399 IC50 = 22 nM T51282 C09MPF 66743431 IC50 = 48 nM T51282 CQ8PM7 66743626 IC50 = 350 nM T51282 CPO12N 66743771 IC50 = 90 nM T51282 C4N6MJ 66743775 IC50 = 35 nM T51282 CZ7V5T 66743809 IC50 = 140 nM T51282 C82RZY 66743831 IC50 = 37 nM T51282 C8F2XJ 66743837 IC50 = 31 nM T51282 CZNY47 66743877 IC50 = 350 nM T51282 CVZ8S6 66744074 IC50 = 100 nM T51282 C64RAW 66744106 IC50 = 2100 nM T51282 CM2XH1 66744214 IC50 = 53 nM T51282 C4T0WG 66744239 IC50 = 100 nM T51282 CE4L0B 66744243 IC50 = 36 nM T51282 CG0V5R 66744251 IC50 = 33 nM T51282 C5F9JE 66906143 IC50 = 6 nM T51282 C37NKO 67129970 IC50 = 8610 nM T51282 CK80LJ 67130050 IC50 > 10000 nM T51282 CV63UL 67240318 IC50 > 10000 nM T51282 C74LIW 67450910 IC50 = 30 nM T51282 CM70FK 68511029 IC50 > 10000 nM T51282 C0UOK4 68512374 IC50 = 610 nM T51282 CLS10P 68513301 IC50 = 11 nM T51282 C5JYB8 68515257 IC50 = 85 nM T51282 CL8SO7 68516150 IC50 = 5100 nM T51282 CP8S0Y 68519792 IC50 = 10 nM T51282 C69OHY 68560854 IC50 = 6 nM T51282 C25MEI 68561431 IC50 = 58 nM T51282 CP1MZ4 68561726 IC50 = 6 nM T51282 CCD89X 68563058 IC50 = 6 nM T51282 C4U2ZW 68565003 IC50 = 33 nM T51282 C0XCY9 68565200 IC50 = 14 nM T51282 CW6BH7 68566254 IC50 = 10 nM T51282 CG7T9J 68566450 IC50 = 11 nM T51282 CQRP72 68567556 IC50 = 13 nM T51282 C48EIQ 68568011 IC50 = 4 nM T51282 C7GRV2 68755406 IC50 > 10000 nM T51282 C5DGR9 69036886 IC50 = 10000 nM T51282 CN7WU6 70681396 IC50 = 31010 nM T51282 CB95AF 70683491 IC50 = 59100 nM T51282 CGC72H 70683492 IC50 = 2610 nM T51282 C56GSR 70687744 IC50 > 400000 nM T51282 C8BJC4 70689793 IC50 = 4600 nM T51282 C0GY4P 70689794 IC50 = 2900 nM T51282 CP7N4B 70689795 IC50 = 2460 nM T51282 CVZ96I 70691888 IC50 = 72500 nM T51282 C5YIS3 70691933 IC50 > 400000 nM T51282 C6JEY5 70691934 IC50 = 2600 nM T51282 C15BRD 70691935 IC50 = 2200 nM T51282 C5V6IR 70693983 IC50 = 21500 nM T51282 CFPJ95 71283262 IC50 < 1 nM T51282 CT92OL 71295837 IC50 > 20000 nM T51282 CKT60L 71455860 Ki = 220 nM T51282 C4AP9J 71506045 IC50 < 1 nM T51282 CVZW12 71529762 IC50 < 1 nM T51282 CMY9K6 71607726 IC50 < 1 nM T51282 C8AM1K 71655603 IC50 = 4 nM T51282 C0DL3F 72698602 IC50 = 0.53 nM T51282 CF9PB2 77105902 IC50 = 5800 nM T51282 CTK3L4 77461132 IC50 = 105 nM T51282 C7U4DH 77461136 IC50 = 203 nM T51282 CL6C4U 77461137 IC50 = 140 nM T51282 CSV23A 78673872 IC50 = 32 nM T51282 CC8I0M 86707711 IC50 = 95 nM T51282 C91YAJ 87405083 IC50 = 5200 nM T51282 CMCL21 87405115 IC50 = 430 nM T51282 CV86ES 87405158 IC50 = 140 nM T51282 CJ64UO 87405222 IC50 = 2100 nM T51282 CVXE69 87405226 IC50 = 5200 nM T51282 CSZ1R0 87405236 IC50 = 400 nM T51282 CIMK73 87405291 IC50 = 50 nM T51282 C5GVJ2 87405534 IC50 = 150 nM T51282 CBF43A 87405559 IC50 = 2900 nM T51282 C3JLM0 87405570 IC50 = 60 nM T51282 CB2H3J 87405750 IC50 = 2400 nM T51282 CN78XC 87405776 IC50 = 110 nM T51282 C9MGP8 87405780 IC50 = 570 nM T51282 CV49YW 87405796 IC50 = 3360 nM T51282 CF87VX 87405826 IC50 = 500 nM T51282 CK8BI1 87405909 IC50 = 52200 nM T51282 CGX1F3 87405928 IC50 = 340 nM T51282 CX6L9J 87405953 IC50 = 380 nM T51282 C1NCJ9 87405962 IC50 = 40 nM T51282 C5VFE9 87405965 IC50 = 620 nM T51282 C1HMK3 87406217 IC50 = 29500 nM T51282 C34SGC 87406334 IC50 = 100 nM T51282 CX79WB 87406347 IC50 = 80 nM T51282 CSY87D 87406371 IC50 = 70 nM T51282 C20FIU 87406393 IC50 = 3700 nM T51282 CLK39G 87406409 IC50 = 43 nM T51282 C2XI8F 87406410 IC50 = 30 nM T51282 CD4FH9 87406443 IC50 = 460 nM T51282 CKH3D4 87406530 IC50 = 90 nM T51282 C23ORM 87406786 IC50 = 1400 nM T51282 CL1TA4 87407566 IC50 = 37800 nM T51282 C74KNV 87408321 IC50 = 1300 nM T51282 CK9VP5 87408525 IC50 = 560 nM T51282 CB5A1I 87481281 IC50 = 720 nM T51282 CP26RT 88898804 IC50 = 6400 nM T51282 CG1L7F 88898863 IC50 = 13000 nM T51282 C20UYR 89421099 IC50 = 120 nM T51282 CE52YZ 89421171 IC50 > 50000 nM T51282 CBY10R 89421243 IC50 = 18700 nM T51282 C45QFT 89421265 IC50 = 30000 nM T51282 CM69ZB 89421450 IC50 = 120 nM T51282 C9SB8C 89421561 IC50 = 640 nM T51282 CK4M3W 89424114 IC50 = 1200 nM T51282 C1HW4B 89735655 IC50 = 2300 nM T51282 CXT1G5 90654805 IC50 = 288 nM T51282 C8BCJ5 90654806 IC50 = 350 nM T51282 C14UGJ 90654807 IC50 = 346 nM T51282 CN67RP 91758287 IC50 = 36 nM T51282 C0Y8ZK 91933875 IC50 > 1000 nM T51282 C9R3XZ 102532131 IC50 = 4390 nM T51282 CK4EN8 117078674 IC50 = 30 nM T51282 CC8XM3 117078749 IC50 = 68 nM T51282 CHQV21 117078751 IC50 = 135 nM T51282 C1KLF8 117078758 IC50 = 169 nM T51282 C7ZL3Q 118715599 IC50 = 12 nM T51282 C8T0AY 118715600 IC50 = 39 nM T51282 C2J3YZ 118715601 IC50 = 141 nM T51282 CRG06J 118715602 IC50 = 52 nM T51282 C7WS3V 118715603 IC50 = 233 nM T51282 CQM81J 118715604 IC50 > 1000 nM T51282 CH3ZB0 118732094 IC50 = 3920 nM T51282 CSYA60 118732095 IC50 = 15050 nM T51282 C0K5LC 118732096 IC50 = 5915 nM T51282 C4HM7F 118732099 IC50 = 7628 nM T51282 C41IOQ 118732101 IC50 = 4317 nM T51282 C2R9JZ 118732102 IC50 > 20000 nM T51282 CG1N5B 118753636 IC50 = 32.6 nM T51282 CN8V5D 118875292 IC50 = 190 nM T51282 CPFQ10 118888903 IC50 = 560 nM T51282 CPVX20 118888909 IC50 = 6700 nM T51282 CG8IB3 118888910 IC50 = 290 nM T51282 C7L9DW 118888912 IC50 = 57 nM T51282 CQI01Y 118888915 IC50 = 400 nM T51282 C6P3LQ 118888916 IC50 = 200 nM T51282 CNH3X7 118888917 IC50 = 69 nM T51282 CW7E1Z 118888918 IC50 = 150 nM T51282 CC8U5M 118888921 IC50 = 12 nM T51282 C61BRC 118888929 IC50 = 97 nM T51282 C15LEY 118888939 IC50 = 23 nM T51282 CKL47W 118888940 IC50 = 21 nM T51282 CRUI71 118888941 IC50 = 11 nM T51282 CEQ5D3 118888943 IC50 = 50 nM T51282 CJQA40 122178640 Ki = 7 nM T51282 CK4Q1D 122178641 Ki = 89 nM T51282 C7I5LX 124636147 IC50 = 523 nM T51282 CW2QI4 127044088 IC50 = 2100 nM T51282 C9NL1A 134475022 IC50 = 19 nM T51282 CU2TB7 134823957 IC50 = 190 nM T51282 CDC38O 134823958 IC50 = 280 nM T51282 C54FXD 134957362 IC50 > 10000 nM T51282 CPV59N 135685787 Ki > 4000 nM T51282 CM2UH4 135894362 IC50 = 17 nM T51282 CY19DW 135894364 IC50 = 48 nM T51282 CF1PS8 135934877 Ki > 4000 nM T51282 CXM24U 135971437 IC50 = 9500 nM T51282 C13AFE 135971438 IC50 = 1400 nM T51282 CAH06E 135971439 IC50 = 9800 nM T51282 C9SL8R 135971440 IC50 > 10000 nM T51282 CCO83V 135971441 IC50 = 7600 nM T51282 CTRL59 135976660 Ki > 4000 nM T51282 CZ06UK 136218660 IC50 = 2 nM T51282 CML48X 136218661 IC50 = 1 nM T51282 COB69I 136218662 IC50 < 1 nM T51282 CSL6Q8 136218663 IC50 = 13 nM T51282 CTFJ83 136226213 IC50 = 7 nM T51282 C5EV8A 136240902 IC50 = 15 nM T51282 CX9LB5 136240903 IC50 = 8 nM T51282 CMC58H 136240944 IC50 = 22 nM T51282 C60PRZ 136241012 IC50 = 16 nM T51282 C1Q9YN 136252259 IC50 = 8 nM T51282 C5YBA1 136333907 IC50 = 140 nM T51282 CJC89A 136333957 IC50 = 420 nM T51282 C7C9YU 136333959 IC50 = 340 nM T51282 C0DWL9 136443810 IC50 = 460 nM T51282 C5U1QO 136443811 IC50 = 940 nM T51282 C54RYQ 136443812 IC50 = 1500 nM T51282 C1RSV0 136443837 IC50 = 400 nM T51282 CAD94U 136603177 IC50 = 370 nM T51282 C9XDB3 136603187 IC50 = 1600 nM T51282 CW62YC 136603199 IC50 = 360 nM T51282 CH0RX6 136603202 IC50 = 450 nM T51282 CL03MU 136603207 IC50 = 540 nM T51282 C03JDR 136603225 IC50 = 530 nM T51282 C4MH3J 136603231 IC50 = 170 nM T51282 C2N7TQ 136603234 IC50 = 830 nM T51282 CAFS87 136603251 IC50 = 770 nM T51282 C6W1JC 136603257 IC50 = 1500 nM T51282 CJ85WI 136603266 IC50 = 130 nM T51282 CG60AI 136603274 IC50 = 260 nM T51282 CGQX59 136603283 IC50 = 1600 nM T51282 C7SCF0 136603308 IC50 = 1700 nM T51282 CS14EM 136603316 IC50 = 160 nM T51282 C45UIL 136603324 IC50 = 4.1 nM T51282 C7K6XF 136603348 IC50 = 760 nM T51282 CW3UG2 136603359 IC50 = 1200 nM T51282 C0H1NQ 136603366 IC50 = 270 nM T51282 C32POI 136603384 IC50 = 360 nM T51282 CI4NV9 136603385 IC50 = 370 nM T51282 CM7Q1G 136603409 IC50 = 420 nM T51282 C63PRK 136603411 IC50 = 630 nM T51282 CN82YH 136603424 IC50 = 40 nM T51282 CI4DH7 136603454 IC50 = 160 nM T51282 C3ELG2 136603459 IC50 = 610 nM T51282 C70AJO 136603466 IC50 = 200 nM T51282 CQU73Y 136603469 IC50 = 96 nM T51282 C9H6WP 136603485 IC50 = 2100 nM T51282 CI1E8V 137634241 IC50 = 5780 nM T51282 C7TG3J 137641313 IC50 = 5370.32 nM T51282 CNH56X 137648287 IC50 = 180 nM T51282 C5KB6I 137661818 IC50 = 820 nM T51282 CC73PA 138911338 IC50 = 64 nM T51282 CU4BG8 139030519 IC50 = 1.22 nM T51282 C69TFH 145976093 IC50 = 1.5 nM T51282 C1K6TQ 145976601 IC50 = 240 nM T51282 C5Z6KS 145980871 IC50 > 1000 nM T51282 CXAP05 145982630 Ki = 16 nM T51282 CV38AJ 145983172 Ki = 19 nM T51282 CAJQ81 145983214 Ki = 40 nM T51282 CPL62H 145991717 IC50 > 1000 nM T51282 CUC18Q 145992833 IC50 > 1000 nM T51282 CSU93V 155077019 IC50 = 38 nM T51282 CIK53P 155510829 IC50 = 3 nM T51282 CK0X8P 155511505 IC50 = 139 nM T51282 C7ZE5Q 155511547 IC50 = 340 nM T51282 CKEP96 155512073 IC50 = 220 nM T51282 CH3FV7 155512419 IC50 = 528 nM T51282 C2MD1Q 155513187 IC50 = 14 nM T51282 C85BYR 155514878 IC50 = 670 nM T51282 C49AVE 155517210 IC50 > 10000 nM T51282 CJR09L 155517677 IC50 > 10000 nM T51282 CW92OR 155517870 IC50 = 650 nM T51282 C7JNV6 155518154 IC50 = 160 nM T51282 CSC9D7 155518157 IC50 = 1500 nM T51282 C86HPW 155518524 IC50 = 35000 nM T51282 CMAU36 155518545 IC50 = 18 nM T51282 C8VJ0R 155519127 IC50 = 16000 nM T51282 CSNO68 155519979 IC50 = 445 nM T51282 CRE3V4 155521980 IC50 = 101 nM T51282 CX87AL 155522068 IC50 = 303 nM T51282 CRI75C 155522515 IC50 = 3951 nM T51282 C1GW0T 155522588 IC50 = 1431 nM T51282 C57TCD 155523512 IC50 = 123 nM T51282 C12KNB 155523817 IC50 = 780 nM T51282 CJH7B6 155524106 IC50 > 10000 nM T51282 C5Y7IU 155524764 IC50 = 117 nM T51282 CL5DR0 155525783 IC50 = 20 nM T51282 CF0XQ6 155525891 IC50 = 49 nM T51282 C8DC7J 155526399 IC50 = 46 nM T51282 CZ1Y2X 155526562 IC50 > 10000 nM T51282 C5UDL7 155527182 IC50 = 235 nM T51282 CWA7T8 155527595 IC50 = 183 nM T51282 CI31SP 155527821 IC50 = 210 nM T51282 C35MHA 155528108 IC50 = 1820 nM T51282 C6KQC9 155529602 IC50 = 280 nM T51282 CFW4G8 155530204 IC50 > 10000 nM T51282 CET2B6 155531372 IC50 = 120 nM T51282 CO7Q5Z 155532093 IC50 > 10000 nM T51282 C7F6MP 155532760 IC50 = 67 nM T51282 CS08FU 155533862 IC50 = 160 nM T51282 COLR41 155533909 IC50 = 39 nM T51282 CX86LP 155534718 IC50 = 473 nM T51282 CR6EI1 155535218 IC50 = 3100 nM T51282 C2EJP6 155535544 IC50 = 550 nM T51282 CZ4U1M 155535897 IC50 = 532 nM T51282 COX2T3 155536115 IC50 = 2502 nM T51282 C76VOG 155536890 IC50 = 803 nM T51282 C2CG1A 155537016 IC50 > 10000 nM T51282 CYV7C2 155537163 IC50 = 6443 nM T51282 C8K3XJ 155537606 IC50 = 110 nM T51282 CE8H4O 155537760 IC50 > 10000 nM T51282 C6QM4V 155537815 IC50 > 10000 nM T51282 CL42XY 155537848 IC50 = 802 nM T51282 C6ZB3U 155538076 IC50 = 4400 nM T51282 CJ50ZQ 155538379 IC50 = 17 nM T51282 CDU52V 155538567 IC50 = 520 nM T51282 CO7J3N 155539166 IC50 > 10000 nM T51282 CXP3U1 155539357 IC50 > 10000 nM T51282 CD8N7Z 155541709 IC50 = 460 nM T51282 CLD14S 155542848 IC50 = 240 nM T51282 C1KM6E 155544122 IC50 = 1052 nM T51282 C2VC7N 155544946 IC50 = 6892 nM T51282 CNF7U3 155545164 IC50 > 10000 nM T51282 C1R5IF 155546763 IC50 = 72 nM T51282 CHEF57 155549647 IC50 = 3741 nM T51282 C8U0DB 155550541 IC50 = 1900 nM T51282 CZ5PL2 155552103 IC50 = 143 nM T51282 C2AZ8C 155553393 IC50 = 1700 nM T51282 CXB5H9 155553912 IC50 = 720 nM T51282 CPV5G8 155555193 IC50 = 1038 nM T51282 C14YJN 155555691 IC50 = 95 nM T51282 C04UNO 155556381 IC50 = 310 nM T51282 C2TMB4 155556732 IC50 = 400 nM T51282 CRP51F 155556776 IC50 = 165 nM T51282 C56FHU 155557272 IC50 = 160 nM T51282 C0QTC9 155557377 IC50 = 869 nM T51282 CNH27R 155557555 IC50 = 9400 nM T51282 C64CJZ 155557560 IC50 = 144 nM T51282 CSO32E 155557808 IC50 > 10000 nM T51282 C0C9PZ 155559054 IC50 = 68 nM T51282 C6A4MZ 155560497 IC50 > 10000 nM T51282 CJ1D6M 155560595 IC50 > 10000 nM T51282 CFBY89 155560747 IC50 = 2400 nM T51282 CLE6M4 155561562 IC50 > 10000 nM T51282 CK7IN8 155562339 IC50 = 990 nM T51282 CU8W7G 155564298 IC50 = 1000 nM T51282 CS19LR 155564577 IC50 > 10000 nM T51282 CWI5K3 155564704 IC50 > 10000 nM T51282 CDU87W 155565976 IC50 = 14 nM T51282 CC1IQ5 155566548 IC50 > 10000 nM T51282 CL1MB0 155567304 IC50 = 580 nM T51282 CSQ69A 155567470 IC50 > 10000 nM T51282 CWMC47 155567479 IC50 = 129 nM T51282 C98WUH 155567548 IC50 = 120 nM T51282 CX91DZ 155567940 IC50 = 1600 nM T51282 CT86WS 155568736 IC50 > 10000 nM T51282 D00ERW 44444843 Ki > 9105 nM T51282 D00HVA 11624601 Ki > 9100 nM T51282 D01YWE 25207521 IC50 = 60 nM T51282 D03CPB 60138149 IC50 = 8 nM T51282 D07ADX 54764565 IC50 = 1030 nM T51282 D07UBK 46911016 IC50 = 1690 nM T51282 D07XWC 44477445 IC50 = 260 nM T51282 D0CM6T 11314340 IC50 = 79 nM T51282 D0EU1R 46215815 IC50 = 7943 nM T51282 D0I1FJ 11393719 IC50 = 100 nM T51282 D0J3LR 11634725 Ki = 1400 nM T51282 D0J7YE 17164245 IC50 = 65000 nM T51282 D0L1UK 3064778 Ki = 31.62 nM T51282 D0L2WP 46225540 IC50 = 1580 nM T51282 D0Q0YV 24944925 IC50 = 4897.79 nM T51282 D0Q3NG 11715520 Ki > 9100 nM T51282 D0R3MO 46864283 IC50 = 10 nM T51282 D0S7IE 11658882 Ki > 9100 nM T51282 D0V0KA 24863112 IC50 = 39 nM T51282 D0W7TU 947057 IC50 > 50000 nM T02024 D06IAR 60961 Ki > 100000 nM T02024 CSR10C 510912 IC50 = 55 nM T02024 COJ29X 890649 IC50 = 5600 nM T02024 C7TZ5D 2930546 IC50 = 20300 nM T02024 C70OXL 3006288 Ki = 15400 nM T02024 CF8N3B 3140491 EC50 > 50000 nM T02024 CAY86S 3312427 IC50 = 8600 nM T02024 CIXQ25 6478685 IC50 = 1500 nM T02024 CW62YA 6479888 IC50 = 770 nM T02024 CN29OD 6618978 IC50 > 50000 nM T02024 CLIF21 9842306 IC50 = 38 nM T02024 CM73SE 9858793 IC50 = 46 nM T02024 CGB78L 9880305 IC50 = 55 nM T02024 CW3S9G 9883477 IC50 = 99 nM T02024 CG16TY 9907596 IC50 = 160 nM T02024 C2X6TP 10233633 Ki = 520 nM T02024 C05NVJ 10259194 Ki = 300 nM T02024 CGF36N 10315709 IC50 = 90 nM T02024 C71JXF 10652408 Ki = 260 nM T02024 CLYM27 10746991 Ki = 340 nM T02024 CDT59Z 10841975 Ki = 37970 nM T02024 CT8DX2 11069304 Ki = 890 nM T02024 C17DLS 11828231 Ki = 2300 nM T02024 C54TFI 12093480 IC50 > 1000 nM T02024 C34QTH 15625173 IC50 = 2600 nM T02024 C3DLS6 15625174 IC50 = 3100 nM T02024 CYX2U3 15625175 IC50 = 1100 nM T02024 CD8B6T 15625184 IC50 = 10900 nM T02024 CJI3P1 15625185 IC50 = 22700 nM T02024 C4X0BA 15625186 IC50 = 2600 nM T02024 CESJ49 15625187 IC50 = 2500 nM T02024 CFLV58 15625188 IC50 = 1800 nM T02024 CX1DZ0 15625192 IC50 = 1200 nM T02024 C8FP9H 15625193 IC50 = 940 nM T02024 CP3L1T 15625194 IC50 = 1800 nM T02024 C1N8XS 16007061 IC50 = 37 nM T02024 C4RKU7 16046198 Ki = 20 nM T02024 CKTA70 16484765 IC50 = 6300 nM T02024 CH0R7U 16484780 IC50 = 9900 nM T02024 CN5AB6 16747704 Ki = 23600 nM T02024 CS42ZC 23626089 IC50 = 4100 nM T02024 CJO79M 23644735 Ki = 73 nM T02024 C2NW5X 23648220 Ki = 19 nM T02024 CCN63I 23648221 Ki = 20 nM T02024 CMVH63 23648222 Ki = 7 nM T02024 C0OR1M 23648223 Ki = 45 nM T02024 C5PIF4 23648224 Ki = 45 nM T02024 C90FQM 23648225 Ki = 10 nM T02024 CB35PV 23648226 Ki = 96 nM T02024 CQ90NK 23648227 Ki = 1 nM T02024 CKZT87 23648228 Ki = 66 nM T02024 CBC71W 23648229 Ki = 16 nM T02024 CYG18K 24748985 Ki = 2070 nM T02024 C6M4QN 24748986 Ki = 5000 nM T02024 CK32AR 24749071 Ki = 400 nM T02024 C9E0AU 24749072 Ki = 2830 nM T02024 CO6DB0 25147739 Ki = 350 nM T02024 C09KIE 25181866 Ki = 7800 nM T02024 CND10S 25181867 Ki > 100000 nM T02024 CX5BU0 25181868 Ki = 2300 nM T02024 C68PMG 25181869 Ki = 44000 nM T02024 C5JVN4 25210968 Ki = 20800 nM T02024 CUZT43 25210969 Ki = 10300 nM T02024 CW8I0P 25879063 IC50 = 150 nM T02024 CXM9L0 44367538 IC50 = 150 nM T02024 CZID50 44367579 IC50 = 83 nM T02024 C70YFO 44415246 Ki = 87 nM T02024 CRZW96 44415248 Ki = 20 nM T02024 C16EMS 44433349 IC50 = 67000 nM T02024 CC2UO4 44440695 IC50 = 23600 nM T02024 COQ83H 44578784 IC50 = 23600 nM T02024 C84EYU 44578785 Ki = 660 nM T02024 C8GJB9 44578786 Ki = 520 nM T02024 C9T2EI 44578787 Ki = 820 nM T02024 CIK76G 44578789 Ki > 100000 nM T02024 CEI32X 44589747 Ki = 42800 nM T02024 C2MF0S 44589785 Ki > 100000 nM T02024 CG7WJ4 44589786 Ki = 97300 nM T02024 CVO20H 46839190 Ki = 14000 nM T02024 C3GET9 46839191 Ki = 77 nM T02024 C0SV8O 46839192 Ki = 1500 nM T02024 C1V3CQ 46839320 Ki = 70 nM T02024 C01DSF 46876831 Ki = 660 nM T02024 CG3RM9 46876832 Ki = 330 nM T02024 CIT31Y 46927861 Ki = 300 nM T02024 CXW02B 46927862 Ki = 580 nM T02024 CU4Z3R 49864088 Ki = 17000 nM T02024 CP5HR1 49864089 Ki = 4400 nM T02024 CQ39WM 49864090 Ki = 1200 nM T02024 C76JYP 49864102 Ki = 8200 nM T02024 CN2G3Z 49864103 Ki = 7100 nM T02024 C01GAC 49864104 Ki = 460 nM T02024 CR8E0Z 51351534 Ki = 5 nM T02024 C9YL2W 51351535 Ki = 99 nM T02024 CPY1M0 51351558 Ki = 16 nM T02024 CT64YQ 52905544 Ki = 522 nM T02024 C81NCO 53317433 Ki = 1100 nM T02024 C81TOB 53317434 Ki = 349 nM T02024 C7R4DT 53317435 Ki = 255 nM T02024 CZ4FR9 53317436 Ki = 77 nM T02024 C0MC6P 53320028 Ki = 5550 nM T02024 C64FAH 53320029 Ki = 14200 nM T02024 CQU37F 53320030 Ki = 94 nM T02024 CFO5E7 53320031 Ki = 70 nM T02024 CN32LO 53320311 Ki = 95 nM T02024 CPO0F3 53322659 Ki = 87 nM T02024 CMT39Y 53322660 Ki = 7900 nM T02024 CN6Q8M 53324226 Ki = 1 nM T02024 CC9D8J 53326788 Ki = 13 nM T02024 C39KQY 71716568 Ki = 110 nM T02024 C3M0JK 72163956 IC50 = 105 nM T02024 CNQ2D6 72945146 Ki = 491 nM T02024 C5OJ0X 72945148 Ki = 39 nM T02024 C01HVL 72945149 Ki = 163 nM T02024 C1OVC0 72945150 Ki = 2553 nM T02024 CBPC50 72945349 Ki = 265 nM T02024 C7MJQ5 72945350 Ki = 3771 nM T02024 C9NTH1 72945351 Ki = 132 nM T02024 CVJ0N8 72945352 Ki = 19 nM T02024 CP1I9N 72945353 Ki = 7723 nM T02024 CJ4R8C 72945541 Ki = 2035 nM T02024 C74WCI 72945542 Ki = 3 nM T02024 C7T3HN 72945732 Ki = 5.6 nM T02024 C95BZQ 72947911 Ki = 13 nM T02024 CCVO01 72947912 Ki = 0.6 nM T02024 CB7HG8 72948102 Ki = 63 nM T02024 C4U3OA 72948103 Ki = 82 nM T02024 CX2U3L 72948104 Ki = 70 nM T02024 C3N7OD 72948105 Ki = 876 nM T02024 CZJ5F6 73346517 Ki = 5556 nM T02024 CN5QE0 73346518 Ki = 892 nM T02024 C26EXZ 73349141 IC50 = 558 nM T02024 CAD90T 73349545 Ki = 4362 nM T02024 CD4BY1 73351103 Ki = 4308 nM T02024 CB94EM 73352218 IC50 = 680 nM T02024 CWO9Q0 73352572 Ki = 854 nM T02024 CPS4I8 76309998 Ki = 38 nM T02024 CB2PT6 76309999 Ki = 56 nM T02024 CL42ER 76310000 Ki = 1679 nM T02024 CI1J4W 76310001 Ki = 1017 nM T02024 CEB47C 76310002 Ki = 2811 nM T02024 C3ICR7 76310003 Ki = 906 nM T02024 C7C9FJ 76317234 Ki = 56 nM T02024 CTLJ38 76317235 Ki = 1828 nM T02024 CZ9U2T 76320941 Ki = 733 nM T02024 C7HJC1 76324606 Ki = 259 nM T02024 C0DFQ1 76328163 Ki = 144 nM T02024 CL41TU 76328164 Ki = 5127 nM T02024 C86TRQ 76331843 Ki = 32 nM T02024 CTFG08 76331844 Ki = 2203 nM T02024 C3OVW6 76335415 Ki = 164 nM T02024 CG7Z4S 76335416 Ki = 259 nM T02024 CD9S8B 90663694 Ki = 110 nM T02024 C1GPY5 145952889 IC50 = 11100 nM T02024 CFQ2O9 145954131 IC50 > 30000 nM T02024 C93AKF 145980356 IC50 = 10100 nM T02024 C67YXK 145980711 IC50 = 13200 nM T02024 CWC78S 145983656 IC50 = 4300 nM T02024 C6VP2S 145985880 IC50 > 30000 nM T02024 C5QBJ2 145989469 IC50 = 20400 nM T02024 C20PUW 145990385 IC50 = 7600 nM T02024 CBL59V 145990969 IC50 = 13800 nM T02024 CP42FJ 145991406 IC50 = 7200 nM T02024 D01LDQ 24749070 Ki = 70 nM T02024 D03HDS 6475540 Ki = 520 nM T02024 D07HZQ 444451 Ki = 33 nM T02024 D0A4AL 477579 Ki = 300 nM T02024 D0S4BK 73680 Ki = 100 nM T02024 D0T4UE 44578788 Ki = 18200 nM T02024 D0Z8EV 446541 IC50 = 19 nM T57307 D02RJY 11442891 IC50 = 621 nM T57307 D0E3TC 44259 IC50 = 14.6 nM T57307 D0Q9UX 16718576 IC50 > 10000 nM T57307 D0T3ME 156422 IC50 > 10000 nM T57307 C4EG8R 24993189 IC50 > 10000 nM T57307 CLS29B 46872626 IC50 > 10000 nM T57307 CV63UL 67240318 IC50 > 10000 nM T57307 C1V3NZ 73425588 IC50 = 6.14 nM T57307 CL0YO5 118443595 IC50 = 47 nM T57307 C6B3TD 146014465 IC50 > 10000 nM T57307 C2MD1Q 155513187 IC50 > 10000 nM T57307 C78MZC 155536330 IC50 = 58 nM T57307 D03DZO 11715767 IC50 > 10000 nM T57307 D0N0LN 46908026 IC50 = 43 nM T57307 D0T8NU 16757525 IC50 > 4000 nM T33969 D00AOJ 12620 IC50 > 1000000 nM T33969 D00AXJ 4189 IC50 < 10000 nM T33969 D00BCP 2727 IC50 = 133000 nM T33969 D00BLL 9849808 IC50 = 133000 nM T33969 D00DKK 5282379 IC50 = 37100 nM T33969 D00FGO 460612 IC50 = 93750 nM T33969 D00FGV 2564 IC50 > 1000000 nM T33969 D00IBN 54676228 IC50 = 133000 nM T33969 D00JAU 3749 IC50 = 7310 nM T33969 D00KHM 16362 IC50 < 10000 nM T33969 D00KVO 2082 IC50 = 133000 nM T33969 D00MIN 657298 IC50 = 133000 nM T33969 D00MYQ 4976 IC50 = 128600 nM T33969 D00NKB 5546 IC50 = 133000 nM T33969 D00NNC 3305 IC50 > 1000000 nM T33969 D00SBN 4746 IC50 = 14360 nM T33969 D00USF 5533 IC50 = 90000 nM T33969 D00WAM 3647 IC50 = 133000 nM T33969 D00WCX 39042 IC50 = 180800 nM T33969 D00WUF 5486971 IC50 = 133000 nM T33969 D00XUN 23894 IC50 = 133000 nM T33969 D00YZA 5453 IC50 = 133000 nM T33969 D00ZFP 5870 IC50 > 1000000 nM T33969 D01AJY 2284 IC50 = 133000 nM T33969 D01AZG 5073 IC50 < 10250 nM T33969 D01DBQ 452548 IC50 = 133000 nM T33969 D01FGR 3100 IC50 > 135000 nM T33969 D01GBY 124087 IC50 = 133000 nM T33969 D01JEU 4054 IC50 > 1000000 nM T33969 D01JUF 5775 IC50 > 1000000 nM T33969 D01KHH 2895 IC50 = 107400 nM T33969 D01KKQ 135400182 IC50 = 133000 nM T33969 D01MDT 5487 IC50 = 133000 nM T33969 D01MUR 68844 IC50 = 133000 nM T33969 D01OXI 2578 IC50 = 97210 nM T33969 D01STB 5362129 IC50 = 133000 nM T33969 D01UTL 2995 IC50 = 133000 nM T33969 D01UXC 2249 IC50 = 133000 nM T33969 D01XNB 4594 IC50 = 75000 nM T33969 D01XOD 54897 IC50 = 9155 nM T33969 D01XYJ 35370 IC50 = 133000 nM T33969 D01ZII 2726 IC50 = 90970 nM T33969 D01ZSO 4235 IC50 = 133000 nM T33969 D02AQY 2018 IC50 > 1000000 nM T33969 D02CKX 31072 IC50 > 1000000 nM T33969 D02DGU 444795 IC50 < 10000 nM T33969 D02DPA 2756 IC50 = 133000 nM T33969 D02FCQ 8699 IC50 > 982300 nM T33969 D02FEM 5284447 IC50 = 133000 nM T33969 D02HED 4748 IC50 = 34840 nM T33969 D02KMO 4826 IC50 = 161300 nM T33969 D02LCR 5467 IC50 = 133000 nM T33969 D02LPF 2123 IC50 > 1000000 nM T33969 D02NTO 5510 IC50 < 10320 nM T33969 D02OZE 2724385 IC50 = 264100 nM T33969 D02PAH 2315 IC50 = 69550 nM T33969 D02PWM 3182 IC50 > 1000000 nM T33969 D02STN 132971 IC50 = 133000 nM T33969 D02TJS 54676038 IC50 = 39930 nM T33969 D02TLO 3690 IC50 = 133000 nM T33969 D02VCJ 443944 IC50 > 1000000 nM T33969 D02WFK 6234 IC50 > 1000000 nM T33969 D02YIZ 12560 IC50 = 133000 nM T33969 D02YPG 667484 IC50 = 61610 nM T33969 D02YYF 2431 IC50 > 1000000 nM T33969 D02ZTJ 5339 IC50 = 133000 nM T33969 D03CJL 3168 IC50 < 10000 nM T33969 D03CQE 5379 IC50 = 133000 nM T33969 D03DAP 3356 IC50 = 217600 nM T33969 D03DDR 3034034 IC50 = 98830 nM T33969 D03ELL 2159 IC50 = 133000 nM T33969 D03FLC 3878 IC50 = 133000 nM T33969 D03GCJ 2583 IC50 > 1000000 nM T33969 D03HJK 447043 IC50 = 133000 nM T33969 D03HYX 441335 IC50 = 9300 nM T33969 D03JSJ 446596 IC50 = 133000 nM T33969 D03KOZ 1549120 IC50 = 36800 nM T33969 D03KQF 4011 IC50 = 133000 nM T33969 D03KZM 216237 IC50 = 9990 nM T33969 D03NHW 4583 IC50 = 133000 nM T33969 D03QGM 5355 IC50 = 276200 nM T33969 D03QWT 73303 IC50 = 133000 nM T33969 D03ROX 2369 IC50 > 1000000 nM T33969 D03RTS 2662 IC50 = 133000 nM T33969 D03RZV 5504 IC50 > 1000000 nM T33969 D03TPR 23690433 IC50 < 10000 nM T33969 D03TVW 54120 IC50 = 133000 nM T33969 D03TYI 9433 IC50 = 133000 nM T33969 D03VPC 2754 IC50 = 133000 nM T33969 D03XOC 656583 IC50 = 133000 nM T33969 D03YLZ 27200 IC50 = 133000 nM T33969 D03ZTE 10133 IC50 = 10600 nM T33969 D04AAW 60613 IC50 = 133000 nM T33969 D04ASH 657180 IC50 = 133000 nM T33969 D04DKH 4418 IC50 < 10000 nM T33969 D04EGX 54746 IC50 = 133000 nM T33969 D04EYC 5906 IC50 > 1000000 nM T33969 D04FBR 5281078 IC50 = 76000 nM T33969 D04ITO 6436173 IC50 = 42000 nM T33969 D04JCN 47811 IC50 = 133000 nM T33969 D04JEE 4946 IC50 = 133000 nM T33969 D04JPJ 3950 IC50 = 133000 nM T33969 D04KTZ 6098 IC50 = 41570 nM T33969 D04KYY 135401907 IC50 > 100000 nM T33969 D04MSM 2554 IC50 = 133000 nM T33969 D04NDM 165580 IC50 > 1000000 nM T33969 D04NQI 2165 IC50 = 77760 nM T33969 D04NXQ 51081 IC50 = 133000 nM T33969 D04OSE 4485 IC50 = 18650 nM T33969 D04QLR 3180 IC50 = 275400 nM T33969 D04RGA 5282415 IC50 = 133000 nM T33969 D04TDQ 4544 IC50 = 23910 nM T33969 D04USC 774 IC50 > 1000000 nM T33969 D04VMT 5253 IC50 = 133000 nM T33969 D04WFD 4543 IC50 = 133000 nM T33969 D04XEG 3343 IC50 > 1000000 nM T33969 D04XGT 31593 IC50 = 133000 nM T33969 D04YMH 151166 IC50 = 133000 nM T33969 D04ZAH 43672 IC50 = 197400 nM T33969 D04ZTY 444020 IC50 = 133000 nM T33969 D05AFX 4450 IC50 = 133000 nM T33969 D05ARP 135398740 IC50 = 133000 nM T33969 D05CEU 941361 IC50 < 10000 nM T33969 D05DVP 5717 IC50 = 11100 nM T33969 D05EAM 4735 IC50 = 133000 nM T33969 D05EPM 3292 IC50 > 791900 nM T33969 D05FTJ 4044 IC50 = 133000 nM T33969 D05GJW 20279 IC50 = 133000 nM T33969 D05HPI 16134395 IC50 = 133000 nM T33969 D05HSC 6000 IC50 = 133000 nM T33969 D05JNI 8378 IC50 > 135000 nM T33969 D05KON 3331 IC50 > 1000000 nM T33969 D05LBU 5472 IC50 = 26950 nM T33969 D05LEO 3385 IC50 = 133000 nM T33969 D05LKP 5215 IC50 = 133000 nM T33969 D05LYX 3488 IC50 = 1500 nM T33969 D05MFA 135398741 IC50 = 133000 nM T33969 D05MQK 110635 IC50 = 133000 nM T33969 D05NOS 5568 IC50 = 39010 nM T33969 D05OFX 219078 IC50 = 133000 nM T33969 D05QDC 5284513 IC50 = 38200 nM T33969 D05RHI 6256 IC50 > 1000000 nM T33969 D05UVD 33624 IC50 = 133000 nM T33969 D05VIL 5284594 IC50 = 133000 nM T33969 D05VIX 3463 IC50 = 133000 nM T33969 D05VLS 5090 IC50 = 95360 nM T33969 D05VQI 2893 IC50 = 15030 nM T33969 D05ZGQ 5281070 IC50 = 133000 nM T33969 D05ZIK 4205 IC50 = 133000 nM T33969 D06ABF 3957 IC50 = 12000 nM T33969 D06AEB 3728 IC50 > 1000000 nM T33969 D06BEP 2712 IC50 = 44100 nM T33969 D06BQU 439503 IC50 > 1000000 nM T33969 D06BYV 6839 IC50 > 1000000 nM T33969 D06CTE 57469 IC50 = 133000 nM T33969 D06FDR 135398739 IC50 = 133000 nM T33969 D06FEA 5280360 IC50 > 1000000 nM T33969 D06FZX 2200 IC50 > 1000000 nM T33969 D06GAM 3357 IC50 = 133000 nM T33969 D06GDY 43815 IC50 = 68910 nM T33969 D06HBQ 91610 IC50 = 11600 nM T33969 D06IIB 443943 IC50 < 10000 nM T33969 D06JPB 5280793 IC50 = 75800 nM T33969 D06NXY 5991 IC50 < 10000 nM T33969 D06OIV 5505 IC50 = 133000 nM T33969 D06OMK 445643 IC50 = 7180 nM T33969 D06ORU 2480 IC50 = 487500 nM T33969 D06OVY 5362065 IC50 = 133000 nM T33969 D06PSS 5311309 IC50 = 133000 nM T33969 D06TNL 3278 IC50 = 133000 nM T33969 D06UDG 60846 IC50 = 31070 nM T33969 D06WTZ 53232 IC50 = 19300 nM T33969 D06XAE 1712095 IC50 = 37000 nM T33969 D06XMU 6013 IC50 = 105000 nM T33969 D06YYD 9578005 IC50 = 133000 nM T33969 D06ZII 969472 IC50 = 133000 nM T33969 D06ZUK 3696 IC50 = 133000 nM T33969 D07ABV 468595 IC50 = 8100 nM T33969 D07BCT 36294 IC50 = 133000 nM T33969 D07BSQ 5994 IC50 < 10000 nM T33969 D07CWD 3657 IC50 = 133000 nM T33969 D07DJQ 10219 IC50 = 133000 nM T33969 D07DVK 20469 IC50 = 10300 nM T33969 D07GRH 2749 IC50 = 133000 nM T33969 D07HBX 338 IC50 > 1000000 nM T33969 D07HGR 5362119 IC50 = 133000 nM T33969 D07HVY 64139 IC50 = 133000 nM T33969 D07IEF 2391 IC50 = 56360 nM T33969 D07IPB 454216 IC50 = 24100 nM T33969 D07JGT 4421 IC50 = 133000 nM T33969 D07JJS 5328 IC50 > 1000000 nM T33969 D07JVL 3016 IC50 = 133000 nM T33969 D07KSG 2733526 IC50 < 10000 nM T33969 D07MCK 5147 IC50 > 1000000 nM T33969 D07MOX 439260 IC50 > 1000000 nM T33969 D07MUN 1054 IC50 > 1000000 nM T33969 D07NAJ 8612 IC50 > 1000000 nM T33969 D07ONP 4753 IC50 > 1000000 nM T33969 D07PAO 17134 IC50 > 1000000 nM T33969 D07POC 176870 IC50 < 10000 nM T33969 D07QCE 2265 IC50 = 133000 nM T33969 D07RGW 4060 IC50 > 1000000 nM T33969 D07SJT 6613 IC50 > 1000000 nM T33969 D07SUG 2478 IC50 = 133000 nM T33969 D07TQV 60825 IC50 = 133000 nM T33969 D07UBG 130881 IC50 = 4730 nM T33969 D07UWJ 2442 IC50 = 20270 nM T33969 D07UYO 441401 IC50 = 133000 nM T33969 D07VDZ 5284627 IC50 = 133000 nM T33969 D07VLY 31703 IC50 = 133000 nM T33969 D07WEP 3019 IC50 = 133000 nM T33969 D07XGR 3339 IC50 = 15300 nM T33969 D07XJM 3042 IC50 = 40040 nM T33969 D07XSN 6253 IC50 = 133000 nM T33969 D07YWY 4417 IC50 < 11040 nM T33969 D07ZTO 2370 IC50 > 1000000 nM T33969 D08CDI 208908 IC50 = 6500 nM T33969 D08EBN 41684 IC50 = 133000 nM T33969 D08HQK 5411 IC50 = 512900 nM T33969 D08HUC 3762 IC50 > 1000000 nM T33969 D08HVR 6047 IC50 = 133000 nM T33969 D08HZC 5852 IC50 = 133000 nM T33969 D08HZL 5574 IC50 = 73720 nM T33969 D08IBS 190 IC50 > 1000000 nM T33969 D08IFL 4037 IC50 = 27240 nM T33969 D08IWD 57363 IC50 = 28200 nM T33969 D08JIV 2162 IC50 = 16000 nM T33969 D08JZS 4992 IC50 > 1000000 nM T33969 D08PIQ 6741 IC50 = 33030 nM T33969 D08QCJ 5430 IC50 = 560000 nM T33969 D08QIP 4887 IC50 = 2970 nM T33969 D08QMX 5757 IC50 = 133000 nM T33969 D08ROP 3899 IC50 = 110000 nM T33969 D08USJ 4456 IC50 = 133000 nM T33969 D08VRO 3822 IC50 = 133000 nM T33969 D08VXL 5353788 IC50 = 133000 nM T33969 D08VXO 6834 IC50 > 100000 nM T33969 D08VYV 4168 IC50 = 133000 nM T33969 D08ZEB 2733 IC50 = 133000 nM T33969 D09AMZ 1676 IC50 > 1000000 nM T33969 D09CZA 5282226 IC50 = 43900 nM T33969 D09DHY 6167 IC50 = 133000 nM T33969 D09DWL 5719 IC50 = 133000 nM T33969 D09EGZ 2719 IC50 = 133000 nM T33969 D09ELP 153994 IC50 = 36350 nM T33969 D09FJB 5503 IC50 = 285700 nM T33969 D09GOS 2812 IC50 < 10000 nM T33969 D09GYT 6082 IC50 > 1000000 nM T33969 D09HNR 3002190 IC50 = 30000 nM T33969 D09HVL 16129704 IC50 = 133000 nM T33969 D09IOI 2170 IC50 = 133000 nM T33969 D09IPV 28417 IC50 < 10000 nM T33969 D09JUG 60490 IC50 = 133000 nM T33969 D09LNI 3365 IC50 = 133000 nM T33969 D09LWS 150311 IC50 = 56000 nM T33969 D09LZT 72287 IC50 = 127000 nM T33969 D09MGR 123619 IC50 = 45000 nM T33969 D09NIA 2732 IC50 = 133000 nM T33969 D09PNY 5593 IC50 = 150900 nM T33969 D09QBG 9854012 IC50 > 1000000 nM T33969 D09QEI 4740 IC50 = 133000 nM T33969 D09RHQ 175805 IC50 = 646400 nM T33969 D09TBD 5344 IC50 = 133000 nM T33969 D09UZO 667490 IC50 = 133000 nM T33969 D09WEJ 2446 IC50 = 133000 nM T33969 D09XQF 3767 IC50 = 133000 nM T33969 D09XZB 123631 IC50 = 10900 nM T33969 D0A0OO 65016 IC50 = 44800 nM T33969 D0A1PX 3394 IC50 = 724700 nM T33969 D0A2ZX 4173 IC50 = 133000 nM T33969 D0A5SE 134018 IC50 = 42900 nM T33969 D0A8XN 3869 IC50 = 649100 nM T33969 D0A9YA 6918296 IC50 = 29800 nM T33969 D0AA2D 2378 IC50 = 27100 nM T33969 D0AD5C 41774 IC50 = 133000 nM T33969 D0AN7B 896 IC50 = 133000 nM T33969 D0AO5H 5578 IC50 = 133000 nM T33969 D0AP9T 53025 IC50 = 133000 nM T33969 D0AR3J 439501 IC50 > 1000000 nM T33969 D0AV3G 3151 IC50 = 133000 nM T33969 D0AZ3C 5291 IC50 < 10000 nM T33969 D0B0CP 667467 IC50 = 27470 nM T33969 D0B1IP 5282375 IC50 = 133000 nM T33969 D0B2GI 3476 IC50 < 10000 nM T33969 D0B2UZ 4917 IC50 < 10000 nM T33969 D0B3HD 2519 IC50 = 133000 nM T33969 D0B5MP 135398513 IC50 = 133000 nM T33969 D0B6TW 135403647 IC50 = 133000 nM T33969 D0B7EB 36462 IC50 = 133000 nM T33969 D0B7NG 2725 IC50 = 133000 nM T33969 D0B7YT 3000322 IC50 > 1000000 nM T33969 D0B8UJ 3011155 IC50 = 133000 nM T33969 D0B8WN 3001055 IC50 > 1000000 nM T33969 D0B9GH 2882 IC50 > 1000000 nM T33969 D0BA6T 38853 IC50 > 1000000 nM T33969 D0BA9U 13109 IC50 = 133000 nM T33969 D0BM5G 5381 IC50 = 133000 nM T33969 D0C0SK 4993 IC50 = 200100 nM T33969 D0C1BG 157355 IC50 > 1000000 nM T33969 D0C1WH 3902 IC50 = 225000 nM T33969 D0C3YQ 23662354 IC50 = 133000 nM T33969 D0C4RB 36314 IC50 = 15000 nM T33969 D0C4YC 4075 IC50 = 381000 nM T33969 D0C6NM 5311221 IC50 = 12900 nM T33969 D0C8EU 5394 IC50 = 133000 nM T33969 D0CF2Q 26879 IC50 > 1000000 nM T33969 D0CL9S 159269 IC50 = 133000 nM T33969 D0CS2F 3955 IC50 = 67000 nM T33969 D0CT9C 2907 IC50 = 133000 nM T33969 D0CW1P 9782 IC50 = 133000 nM T33969 D0CZ1Q 5311067 IC50 = 16420 nM T33969 D0D0BE 28061 IC50 = 133000 nM T33969 D0D0ZD 441314 IC50 = 133000 nM T33969 D0D1AL 3559 IC50 = 22760 nM T33969 D0D1SG 5755 IC50 = 91470 nM T33969 D0D2VS 60198 IC50 = 90000 nM T33969 D0D4JO 6917864 IC50 = 133000 nM T33969 D0D5GD 3373 IC50 > 100000 nM T33969 D0D5GG 4723 IC50 = 133000 nM T33969 D0D7KC 5488548 IC50 = 133000 nM T33969 D0D7LA 4091 IC50 = 133000 nM T33969 D0D8XY 5311010 IC50 = 133000 nM T33969 D0D9FV 4601 IC50 > 1000000 nM T33969 D0DJ1B 156391 IC50 = 133000 nM T33969 D0E0CT 5573 IC50 < 10000 nM T33969 D0E0LQ 941651 IC50 = 30400 nM T33969 D0E0SW 53708 IC50 = 133000 nM T33969 D0E1SW 1986 IC50 = 133000 nM T33969 D0E1XL 5284583 IC50 = 133000 nM T33969 D0E3OF 54678486 IC50 = 115300 nM T33969 D0E6OC 5282230 IC50 = 41500 nM T33969 D0E6XR 3062316 IC50 < 10000 nM T33969 D0E6YQ 1935 IC50 = 133000 nM T33969 D0E7PQ 5311 IC50 = 133000 nM T33969 D0E8CI 5282443 IC50 = 290800 nM T33969 D0EG1I 9926791 IC50 = 133000 nM T33969 D0EJ6O 2763 IC50 = 133000 nM T33969 D0ES1Q 6918289 IC50 = 2690 nM T33969 D0EV8E 3198 IC50 < 10000 nM T33969 D0F2PO 4828 IC50 = 133000 nM T33969 D0F6EO 33613 IC50 = 133000 nM T33969 D0F7CS 6758 IC50 = 8000 nM T33969 D0F8RA 2153 IC50 = 133000 nM T33969 D0F9GE 3108 IC50 = 4000 nM T33969 D0FA2O 5585 IC50 > 525100 nM T33969 D0FM2P 82153 IC50 = 133000 nM T33969 D0FN7J 4107 IC50 > 1000000 nM T33969 D0FT4R 107706 IC50 = 142200 nM T33969 D0FX2Q 6324616 IC50 = 6300 nM T33969 D0G3DL 135398735 IC50 = 11300 nM T33969 D0G3SH 31401 IC50 < 10000 nM T33969 D0G4OD 54686904 IC50 = 133000 nM T33969 D0G5AG 104762 IC50 = 133000 nM T33969 D0G5QB 51263 IC50 > 135000 nM T33969 D0G5UB 2161 IC50 = 104000 nM T33969 D0G7FJ 54677470 IC50 = 77500 nM T33969 D0G8NN 119570 IC50 = 133000 nM T33969 D0G9IU 135403821 IC50 = 9910 nM T33969 D0G9YH 2179 IC50 = 133000 nM T33969 D0GL7U 6230 IC50 = 18460 nM T33969 D0GU4K 135413536 IC50 = 133000 nM T33969 D0GY5Z 2244 IC50 = 133000 nM T33969 D0H0HJ 19493 IC50 > 1000000 nM T33969 D0H0KB 5070 IC50 = 133000 nM T33969 D0H0ND 54454 IC50 < 10000 nM T33969 D0H1GJ 5325 IC50 > 1000000 nM T33969 D0H1YQ 71764 IC50 = 133000 nM T33969 D0H2DQ 4912 IC50 > 1000000 nM T33969 D0H2SY 4633 IC50 = 309100 nM T33969 D0H3HM 60795 IC50 = 133000 nM T33969 D0H3TD 104838 IC50 > 1000000 nM T33969 D0H3WI 37542 IC50 = 133000 nM T33969 D0H4JM 8969 IC50 = 254000 nM T33969 D0H6QU 6005 IC50 = 133000 nM T33969 D0H8FH 3702 IC50 = 144700 nM T33969 D0H9ZQ 131204 IC50 > 1000000 nM T33969 D0HQ6N 1201549 IC50 = 188600 nM T33969 D0I0EG 44093 IC50 = 133000 nM T33969 D0I0RJ 16231 IC50 > 1000000 nM T33969 D0I2MK 4171 IC50 = 133000 nM T33969 D0I4DQ 5280723 IC50 = 133000 nM T33969 D0I6IB 54677971 IC50 = 133000 nM T33969 D0I7SZ 54892 IC50 = 15500 nM T33969 D0I8DD 6914273 IC50 = 145500 nM T33969 D0I8FI 3779 IC50 > 986200 nM T33969 D0IT2G 5743 IC50 = 101700 nM T33969 D0IT2X 2581 IC50 = 133000 nM T33969 D0IX6I 222786 IC50 = 108100 nM T33969 D0J0ZS 3446 IC50 > 1000000 nM T33969 D0J1MI 4030 IC50 = 133000 nM T33969 D0J1VY 5281081 IC50 = 55600 nM T33969 D0J2KV 4932 IC50 = 53700 nM T33969 D0J2MJ 26758 IC50 = 133000 nM T33969 D0J4GO 3038 IC50 > 919100 nM T33969 D0J4JM 5770 IC50 = 8350 nM T33969 D0J5DC 2796 IC50 = 60000 nM T33969 D0J7RK 36811 IC50 > 100000 nM T33969 D0J9XZ 41781 IC50 = 130700 nM T33969 D0JC9N 60164 IC50 = 133000 nM T33969 D0JO7Y 104741 IC50 = 133000 nM T33969 D0JV4Q 3002820 IC50 = 9650 nM T33969 D0JY3V 107751 IC50 = 20300 nM T33969 D0K0OZ 5702160 IC50 = 133000 nM T33969 D0K0TC 68617 IC50 = 29340 nM T33969 D0K0VO 5639 IC50 < 11300 nM T33969 D0K1XK 3637 IC50 > 1000000 nM T33969 D0K3MC 3947 IC50 = 133000 nM T33969 D0K3QS 6442177 IC50 = 2000 nM T33969 D0K5CB 2083 IC50 = 133000 nM T33969 D0K6GZ 60464 IC50 = 133000 nM T33969 D0K7HU 6918155 IC50 = 133000 nM T33969 D0K7WK 4595 IC50 = 133000 nM T33969 D0K8KX 5280343 IC50 = 133000 nM T33969 D0KD1U 4883 IC50 > 1000000 nM T33969 D0KG3R 9875401 IC50 = 133000 nM T33969 D0KR2J 135398508 IC50 = 133000 nM T33969 D0KR5B 5754 IC50 = 251700 nM T33969 D0L0SW 6957673 IC50 = 234800 nM T33969 D0L2MX 2343 IC50 = 57430 nM T33969 D0L3DK 6918537 IC50 = 133000 nM T33969 D0L4HY 5702063 IC50 = 343700 nM T33969 D0L5RW 65015 IC50 = 133000 nM T33969 D0L5WM 2157 IC50 < 10000 nM T33969 D0L6DA 119607 IC50 = 133000 nM T33969 D0L7FM 4911 IC50 = 133000 nM T33969 D0L9ZR 4891 IC50 = 60270 nM T33969 D0M2MR 3475 IC50 = 133000 nM T33969 D0M3QP 441207 IC50 < 10000 nM T33969 D0M4VM 5320 IC50 > 1000000 nM T33969 D0M4YC 3114 IC50 = 133000 nM T33969 D0M5JI 9560989 IC50 = 133000 nM T33969 D0M5OC 5484727 IC50 = 133000 nM T33969 D0M6DO 2145 IC50 = 133000 nM T33969 D0M8RC 5403 IC50 = 133000 nM T33969 D0M8VE 71360 IC50 = 23400 nM T33969 D0M9BW 68911 IC50 = 133000 nM T33969 D0M9DC 4614 IC50 = 133000 nM T33969 D0MA9N 2955 IC50 = 133000 nM T33969 D0ML1F 60871 IC50 = 46000 nM T33969 D0MP5H 2966 IC50 > 951800 nM T33969 D0MY8N 5280489 IC50 < 10000 nM T33969 D0N0EQ 19649 IC50 > 1000000 nM T33969 D0N0RU 82146 IC50 = 133000 nM T33969 D0N0TZ 60606 IC50 = 72000 nM T33969 D0N1FS 26248 IC50 = 133000 nM T33969 D0N3PE 3518 IC50 > 1000000 nM T33969 D0N3VR 71616 IC50 = 133000 nM T33969 D0N4OW 644077 IC50 = 133000 nM T33969 D0N5HJ 5462501 IC50 = 133000 nM T33969 D0N5YA 65981 IC50 = 22000 nM T33969 D0N6RF 65999 IC50 = 16200 nM T33969 D0NG7O 60857 IC50 = 133000 nM T33969 D0NJ3V 4680 IC50 < 10000 nM T33969 D0NR6S 3002977 IC50 = 110000 nM T33969 D0NS6H 3152 IC50 = 78000 nM T33969 D0NW3X 71329 IC50 = 708400 nM T33969 D0O1WX 2764 IC50 = 133000 nM T33969 D0O2EM 4463 IC50 = 294600 nM T33969 D0O2SR 47528 IC50 = 133000 nM T33969 D0O2WB 4991 IC50 > 1000000 nM T33969 D0O3OS 104850 IC50 < 10000 nM T33969 D0O4SE 5479 IC50 = 133000 nM T33969 D0O5FY 441130 IC50 = 133000 nM T33969 D0O5WP 148124 IC50 = 41000 nM T33969 D0O5YZ 71698 IC50 = 35870 nM T33969 D0O6IZ 4436 IC50 > 1000000 nM T33969 D0O6SX 3658 IC50 = 72910 nM T33969 D0OB1J 39186 IC50 = 133000 nM T33969 D0OT0O 44561 IC50 = 133000 nM T33969 D0P0HB 2761171 IC50 > 1000000 nM T33969 D0P0HT 9878 IC50 = 100900 nM T33969 D0P1UX 5656 IC50 = 133000 nM T33969 D0P1WA 5487427 IC50 > 1000000 nM T33969 D0P5GE 3025 IC50 = 41650 nM T33969 D0P5SA 3372 IC50 = 25820 nM T33969 D0P7JZ 34359 IC50 = 133000 nM T33969 D0P9AC 3675 IC50 > 897200 nM T33969 D0P9RF 5401 IC50 = 133000 nM T33969 D0PG8O 5360515 IC50 > 1000000 nM T33969 D0PQ3G 3440 IC50 = 133000 nM T33969 D0PW7C 51039 IC50 = 133000 nM T33969 D0Q0RC 3290 IC50 = 139200 nM T33969 D0Q2AT 21319 IC50 < 10000 nM T33969 D0Q2ES 7699 IC50 < 10000 nM T33969 D0Q2PE 4539 IC50 = 133000 nM T33969 D0Q2XF 5311027 IC50 = 40400 nM T33969 D0Q3YO 1547484 IC50 = 15700 nM T33969 D0Q4SD 443872 IC50 = 133000 nM T33969 D0Q4XQ 3291 IC50 = 133000 nM T33969 D0Q4YK 4843 IC50 = 133000 nM T33969 D0Q5NX 216326 IC50 = 133000 nM T33969 D0Q5UQ 214348 IC50 = 58400 nM T33969 D0Q6NZ 5281034 IC50 = 48700 nM T33969 D0Q8ZX 2337 IC50 = 133000 nM T33969 D0Q9HF 187 IC50 > 1000000 nM T33969 D0Q9JT 4174 IC50 = 229000 nM T33969 D0QL3P 34312 IC50 = 133000 nM T33969 D0QS1U 10230 IC50 > 1000000 nM T33969 D0R0BX 6604200 IC50 = 133000 nM T33969 D0R0FE 2520 IC50 = 133000 nM T33969 D0R0MW 5329102 IC50 = 45810 nM T33969 D0R0UJ 4688 IC50 > 1000000 nM T33969 D0R1QE 3672 IC50 > 135000 nM T33969 D0R1RS 3715 IC50 = 42000 nM T33969 D0R1WR 4919 IC50 = 133000 nM T33969 D0R2KJ 18381 IC50 < 10000 nM T33969 D0R2KY 9270 IC50 = 62000 nM T33969 D0R3FP 6398764 IC50 = 133000 nM T33969 D0R3QY 5665 IC50 = 133000 nM T33969 D0R4OM 5566 IC50 < 10000 nM T33969 D0R5RR 119182 IC50 = 133000 nM T33969 D0R6BI 3341 IC50 > 1000000 nM T33969 D0R6RO 4184 IC50 = 46820 nM T33969 D0R7HO 2471 IC50 = 133000 nM T33969 D0R8ER 3229 IC50 = 133000 nM T33969 D0R9OH 5329 IC50 = 133000 nM T33969 D0R9VR 9651 IC50 = 133000 nM T33969 D0RD5W 154417 IC50 > 1000000 nM T33969 D0RG3O 174174 IC50 > 135000 nM T33969 D0S1NZ 5310993 IC50 = 133000 nM T33969 D0S3WH 68827 IC50 = 133000 nM T33969 D0S4BR 1349907 IC50 = 133000 nM T33969 D0S5CU 4499 IC50 = 33000 nM T33969 D0S5UH 2794 IC50 = 12900 nM T33969 D0S5WG 3366 IC50 = 133000 nM T33969 D0S6JG 5920 IC50 = 11270 nM T33969 D0S9MC 2789 IC50 = 133000 nM T33969 D0S9SD 60877 IC50 = 133000 nM T33969 D0SH3I 387447 IC50 = 133000 nM T33969 D0SV8E 126941 IC50 = 133000 nM T33969 D0T0KA 4474 IC50 = 7870 nM T33969 D0T0LM 4848 IC50 > 1000000 nM T33969 D0T1LK 4908 IC50 = 32700 nM T33969 D0T2PL 5280453 IC50 = 39700 nM T33969 D0T2XU 4927 IC50 = 133000 nM T33969 D0T3AD 439693 IC50 = 133000 nM T33969 D0T3NY 688020 IC50 = 109500 nM T33969 D0T5WK 4506 IC50 = 133000 nM T33969 D0T7OW 681 IC50 > 1000000 nM T33969 D0T7US 5281037 IC50 = 133000 nM T33969 D0T8GD 89594 IC50 = 133000 nM T33969 D0T8VY 71771 IC50 = 105000 nM T33969 D0T9DT 2140 IC50 = 133000 nM T33969 D0T9TJ 3034010 IC50 = 133000 nM T33969 D0TG1H 3033 IC50 = 44000 nM T33969 D0TR5X 3386 IC50 = 133000 nM T33969 D0TZ1G 4914 IC50 > 1000000 nM T33969 D0U0KW 208902 IC50 = 85000 nM T33969 D0U1OE 5452 IC50 = 24330 nM T33969 D0U1OM 60726 IC50 = 133000 nM T33969 D0U2CV 5531 IC50 = 627800 nM T33969 D0U2JP 4369359 IC50 = 133000 nM T33969 D0U2OO 2477 IC50 = 59630 nM T33969 D0U4CE 104865 IC50 = 22000 nM T33969 D0U4UQ 3639 IC50 = 133000 nM T33969 D0U5CE 1548943 IC50 < 10000 nM T33969 D0U5GB 92727 IC50 = 17300 nM T33969 D0U5QK 1983 IC50 = 133000 nM T33969 D0U5RT 4909 IC50 = 133000 nM T33969 D0U5SI 4913 IC50 = 133000 nM T33969 D0U6LM 4192 IC50 = 41700 nM T33969 D0U7GK 5426 IC50 > 1000000 nM T33969 D0U8UV 10660 IC50 = 133000 nM T33969 D0UA0I 28693 IC50 < 10000 nM T33969 D0UF6M 9568512 IC50 = 133000 nM T33969 D0UL2L 54690031 IC50 = 7560 nM T33969 D0UM7O 3821 IC50 = 133000 nM T33969 D0V0LB 6058 IC50 = 331000 nM T33969 D0V4QS 135398745 IC50 = 54570 nM T33969 D0V7CF 5362440 IC50 = 21200 nM T33969 D0V7XF 55483 IC50 > 1000000 nM T33969 D0V8QT 2708 IC50 = 133000 nM T33969 D0V9BD 2375 IC50 = 29300 nM T33969 D0V9YR 5327 IC50 > 1000000 nM T33969 D0VM2L 68740 IC50 = 133000 nM T33969 D0VP1V 11434515 IC50 = 127100 nM T33969 D0VR7W 9571107 IC50 > 1000000 nM T33969 D0VT8P 3324 IC50 = 133000 nM T33969 D0W0BF 2187 IC50 = 133000 nM T33969 D0W5HK 216239 IC50 < 10000 nM T33969 D0W6DY 3103 IC50 = 508800 nM T33969 D0W9LX 2585 IC50 = 133000 nM T33969 D0WE3O 5288826 IC50 > 135000 nM T33969 D0WI3T 441243 IC50 = 2900 nM T33969 D0WN0U 3333 IC50 = 69700 nM T33969 D0WS1X 6915944 IC50 = 133000 nM T33969 D0WV3U 4893 IC50 = 133000 nM T33969 D0X0RI 4178 IC50 = 133000 nM T33969 D0X2DK 4768 IC50 > 100000 nM T33969 D0X2MB 4631 IC50 > 1000000 nM T33969 D0X3FX 5284596 IC50 = 133000 nM T33969 D0X4RN 3676 IC50 = 133000 nM T33969 D0X4ZR 444 IC50 > 1000000 nM T33969 D0X5SD 3117 IC50 < 10000 nM T33969 D0X5XU 451668 IC50 = 133000 nM T33969 D0X6GN 444025 IC50 = 40400 nM T33969 D0X6IU 5959 IC50 = 133000 nM T33969 D0X7DE 4449 IC50 = 6100 nM T33969 D0X7JN 5280980 IC50 > 1000000 nM T33969 D0X7KZ 6918182 IC50 = 133000 nM T33969 D0X7XG 3000226 IC50 = 10100 nM T33969 D0X9RG 5361092 IC50 = 133000 nM T33969 D0X9ZC 47965 IC50 = 133000 nM T33969 D0XB8P 247 IC50 > 1000000 nM T33969 D0XF8W 1046 IC50 = 133000 nM T33969 D0Y0JH 5161 IC50 > 1000000 nM T33969 D0Y0SW 3397 IC50 = 60780 nM T33969 D0Y2CJ 4201 IC50 = 133000 nM T33969 D0Y2LR 3162 IC50 > 1000000 nM T33969 D0Y2YP 15209 IC50 = 71190 nM T33969 D0Y3KG 3121 IC50 > 1000000 nM T33969 D0Y3MO 37768 IC50 = 133000 nM T33969 D0Y4DY 5709 IC50 > 796100 nM T33969 D0Y4JJ 2351 IC50 < 16460 nM T33969 D0Y5DO 2771 IC50 = 133000 nM T33969 D0Y5UG 2160 IC50 = 133000 nM T33969 D0Y7EM 3332 IC50 = 133000 nM T33969 D0Y7IU 5281004 IC50 = 46000 nM T33969 D0Y7PG 4659569 IC50 < 33920 nM T33969 D0Y7RW 4763 IC50 > 135000 nM T33969 D0Y7ZU 135398738 IC50 = 133000 nM T33969 D0Y9LL 42884 IC50 = 133000 nM T33969 D0YG7M 3827 IC50 = 738400 nM T33969 D0YV1Q 6032 IC50 = 133000 nM T33969 D0Z0DW 135398658 IC50 > 1000000 nM T33969 D0Z1FX 5756 IC50 > 1000000 nM T33969 D0Z1RV 135398737 IC50 = 75140 nM T33969 D0Z1ZM 84029 IC50 = 133000 nM T33969 D0Z3DY 2333 IC50 = 17500 nM T33969 D0Z4EI 55245 IC50 = 2020 nM T33969 D0Z4SB 3478 IC50 = 133000 nM T33969 D0Z4UN 6509979 IC50 = 10000 nM T33969 D0Z4ZT 68873 IC50 = 16400 nM T33969 D0Z5BC 5634 IC50 = 133000 nM T33969 D0Z5IU 1548887 IC50 = 226000 nM T33969 D0Z5OE 4211 IC50 < 10000 nM T33969 D0Z6UC 5358 IC50 = 133000 nM T33969 D0Z7KE 3784 IC50 = 28000 nM T33969 D0Z7ZM 135398744 IC50 = 16430 nM T33969 D0Z8EX 18283 IC50 = 133000 nM T33969 D0Z9QR 24066 IC50 = 133000 nM T33969 D0ZB7K 5735 IC50 = 133000 nM T33969 D0ZS8P 2801 IC50 = 133000 nM T33969 D0ZU9R 392622 IC50 = 1740 nM T33969 D00GEG 5745207 IC50 = 174700 nM T33969 D00QAR 5904 IC50 < 10000 nM T33969 D00QKI 9865554 IC50 < 10000 nM T33969 D00TIG 6917964 IC50 = 9340 nM T33969 D01LXD 9843750 IC50 = 471900 nM T33969 D02AIN 122678117 IC50 = 74000 nM T33969 D02EVF 6112 IC50 > 1000000 nM T33969 D02JUW 460 IC50 > 1000000 nM T33969 D02NNV 3038525 IC50 < 10000 nM T33969 D02OJC 128919 IC50 = 117100 nM T33969 D02YEY 128268 IC50 = 23030 nM T33969 D04FNQ 56237 IC50 = 14390 nM T33969 D04GZS 137994 IC50 > 1000000 nM T33969 D05JET 60511 IC50 = 288100 nM T33969 D06CCR 50313 IC50 > 1000000 nM T33969 D06GRK 4494 IC50 < 10000 nM T33969 D06RYY 9843028 IC50 = 490000 nM T33969 D07EFM 2230 IC50 > 1000000 nM T33969 D08YWK 6436 IC50 = 133000 nM T33969 D09YDM 24360 IC50 = 133000 nM T33969 D0B1FE 3194 IC50 < 10000 nM T33969 D0CE0O 11513676 IC50 = 110 nM T33969 D0E3TC 44259 IC50 = 18700 nM T33969 D0G7UX 5284373 IC50 = 500 nM T33969 D0GC5H 123879 IC50 = 62400 nM T33969 D0H0YD 32798 IC50 = 8500 nM T33969 D0I8FV 5567 IC50 = 19700 nM T33969 D0K5HI 5311424 IC50 < 10000 nM T33969 D0KE4Z 5310954 IC50 > 1000000 nM T33969 D0L1VF 32343 IC50 < 10000 nM T33969 D0P6DJ 151194 IC50 < 10000 nM T33969 D0Q7QY 53359 IC50 = 185300 nM T33969 D0Q9CY 9915743 IC50 = 25000 nM T33969 D0S0EQ 9951066 IC50 < 10000 nM T33969 D0S6TK 11213558 IC50 = 196600 nM T33969 D0SD9V 53276 IC50 = 35500 nM T33969 D0TO2R 30751 IC50 = 133000 nM T33969 D0VG0D 11977753 IC50 = 7900 nM T33969 D0W8XT 60663 IC50 = 25000 nM T33969 D0X8ED 2327 IC50 = 116600 nM T33969 D0Y1FO 472335 IC50 = 133000 nM T33969 D00CCI 39941 IC50 = 175000 nM T33969 D00UEQ 9840324 IC50 = 11800 nM T33969 D01PIL 54477 IC50 < 10000 nM T33969 D01VAB 2119 IC50 = 133000 nM T33969 D02FNU 56971 IC50 = 31170 nM T33969 D02LHR 33625 IC50 = 109000 nM T33969 D03BOZ 3342298 IC50 = 23360 nM T33969 D03DRW 9803778 IC50 < 13510 nM T33969 D03GFC 16741245 IC50 < 12850 nM T33969 D03JPH 54677972 IC50 = 133000 nM T33969 D04BQR 4342 IC50 = 133000 nM T33969 D04EEU 53001 IC50 > 1000000 nM T33969 D05JQF 6917939 IC50 < 10000 nM T33969 D05RUM 15387 IC50 = 133000 nM T33969 D06ABW 2788 IC50 = 133000 nM T33969 D06BPG 4528 IC50 > 1000000 nM T33969 D06LGC 9906649 IC50 > 1000000 nM T33969 D07XPE 8249 IC50 = 133000 nM T33969 D08DKA 93504 IC50 = 353300 nM T33969 D08SOF 5405 IC50 < 17470 nM T33969 D09JVV 5983 IC50 > 1000000 nM T33969 D09PTA 132228 IC50 < 10000 nM T33969 D09WFI 14296 IC50 > 1000000 nM T33969 D0B9GM 4622 IC50 > 1000000 nM T33969 D0C0JT 4495 IC50 = 133000 nM T33969 D0C1XS 5365247 IC50 = 229700 nM T33969 D0C5PA 183812 IC50 < 10000 nM T33969 D0F7TV 65888 IC50 = 304900 nM T33969 D0FX4J 5387 IC50 = 315300 nM T33969 D0G9ZW 54676478 IC50 = 133000 nM T33969 D0J9GD 64715 IC50 = 27000 nM T33969 D0N0LB 6103 IC50 > 1000000 nM T33969 D0O2IE 4754 IC50 = 133000 nM T33969 D0O6AQ 6450546 IC50 < 10000 nM T33969 D0O8OB 3783 IC50 = 572500 nM T33969 D0OS6O 60149 IC50 = 82700 nM T33969 D0P1JI 312145 IC50 = 13600 nM T33969 D0S6QR 214350 IC50 = 133000 nM T33969 D0S8YL 3969 IC50 < 10740 nM T33969 D0T1RG 216235 IC50 = 12600 nM T33969 D0X7HV 177852 IC50 = 21390 nM T33969 D0Y0GG 72014 IC50 = 244400 nM T33969 D0Y2HR 2247 IC50 < 10000 nM T33969 D0Y4FL 6915744 IC50 = 133000 nM T33969 D0Y8UB 82148 IC50 = 133000 nM T33969 D0Z0CH 3033962 IC50 = 55750 nM T33969 CDF6T9 85 IC50 > 1000000 nM T33969 CPF48I 904 IC50 > 1000000 nM T33969 CBM59A 989 IC50 > 1000000 nM T33969 CQG8W1 1309 IC50 = 65640 nM T33969 C6JB0E 1599 IC50 > 1000000 nM T33969 CF6O0D 1985 IC50 > 1000000 nM T33969 C26XBL 2017 IC50 = 43480 nM T33969 C8D9QE 2031 IC50 = 158400 nM T33969 C5IQN3 2075 IC50 > 1000000 nM T33969 C9ARM2 2178 IC50 > 1000000 nM T33969 C85KQB 2202 IC50 = 133000 nM T33969 CXUC05 2215 IC50 = 390900 nM T33969 CK37XY 2311 IC50 = 74860 nM T33969 CI74WY 2450 IC50 = 133000 nM T33969 CIT06W 2482 IC50 = 181100 nM T33969 C45PUM 2551 IC50 > 1000000 nM T33969 CC7D8I 2723 IC50 = 129900 nM T33969 CPJ0C2 2747 IC50 = 133000 nM T33969 C36WOC 2800 IC50 < 10000 nM T33969 C7CT6M 2804 IC50 = 133000 nM T33969 CH93VI 2817 IC50 = 356700 nM T33969 CLSX94 2975 IC50 = 202200 nM T33969 CJOC76 3023 IC50 = 387900 nM T33969 CJTA06 3081 IC50 > 1000000 nM T33969 CJ0B9F 3158 IC50 = 133000 nM T33969 C0H8GR 3191 IC50 = 133000 nM T33969 CEXU05 3383 IC50 = 133000 nM T33969 CYCX32 3420 IC50 < 13340 nM T33969 CR0M3G 3474 IC50 < 14930 nM T33969 CPER58 3516 IC50 > 1000000 nM T33969 COSX53 3519 IC50 = 133000 nM T33969 C7HRW8 3609 IC50 > 1000000 nM T33969 CUT30Q 3616 IC50 > 1000000 nM T33969 CHV5M7 3634 IC50 = 29800 nM T33969 CO2Y3R 3698 IC50 = 133000 nM T33969 C4ZJT8 3730 IC50 = 133000 nM T33969 CY4WG9 3793 IC50 = 18000 nM T33969 C9LCD8 3823 IC50 = 3400 nM T33969 C2KJI7 3883 IC50 = 133000 nM T33969 CY18JF 4059 IC50 > 1000000 nM T33969 C8F4XW 4065 IC50 > 1000000 nM T33969 C68LHN 4086 IC50 > 1000000 nM T33969 CV0F2R 4098 IC50 > 1000000 nM T33969 C12UDR 4411 IC50 = 133000 nM T33969 CD0SK3 4454 IC50 > 1000000 nM T33969 CQ72GP 4511 IC50 = 184500 nM T33969 C60PHU 4567 IC50 = 280000 nM T33969 CG18LW 4621 IC50 < 10000 nM T33969 CW2QL9 4686 IC50 = 33560 nM T33969 CX8H9B 4782 IC50 > 1000000 nM T33969 CZF18J 4811 IC50 > 1000000 nM T33969 CQI08L 4814 IC50 = 441000 nM T33969 C98DJE 4819 IC50 > 1000000 nM T33969 C8VXJ6 4888 IC50 = 133000 nM T33969 C5IOL8 4910 IC50 < 13190 nM T33969 C93BJO 5039 IC50 = 133000 nM T33969 CXQ02H 5104 IC50 > 1000000 nM T33969 C3L0UM 5315 IC50 > 1000000 nM T33969 CWVF28 5323 IC50 > 1000000 nM T33969 C5N0SU 5334 IC50 = 133000 nM T33969 CSNK90 5424 IC50 > 1000000 nM T33969 C2I7CF 5443 IC50 > 1000000 nM T33969 C48GPY 5475 IC50 = 133000 nM T33969 C7SCP4 5478 IC50 > 1000000 nM T33969 C1EYR7 5497 IC50 = 133000 nM T33969 C37UQK 5606 IC50 > 1000000 nM T33969 C8Y9ZN 5641 IC50 > 1000000 nM T33969 C78PXT 5794 IC50 < 10000 nM T33969 CG8V9E 5917 IC50 > 1000000 nM T33969 CH13XE 6034 IC50 = 478500 nM T33969 C78ENM 6077 IC50 = 111600 nM T33969 C2U1WA 6216 IC50 = 133000 nM T33969 C59UQE 6279 IC50 = 15700 nM T33969 CL53OW 6461 IC50 > 1000000 nM T33969 C1IO8J 6634 IC50 > 1000000 nM T33969 CZ2C9Y 6857 IC50 = 68680 nM T33969 C3H5DF 7172 IC50 > 1000000 nM T33969 CJ7PK9 8574 IC50 > 1000000 nM T33969 CR6HO1 8593 IC50 = 695300 nM T33969 C40HCL 8987 IC50 = 69260 nM T33969 CTEL83 9279 IC50 = 291300 nM T33969 CC09DB 9703 IC50 = 133000 nM T33969 CILW30 10718 IC50 > 1000000 nM T33969 CO1I7C 11080 IC50 = 60000 nM T33969 CMU2P6 11683 IC50 < 10000 nM T33969 C2QS4E 12478 IC50 > 1000000 nM T33969 C2J7BV 12947 IC50 = 133000 nM T33969 CVJ2X3 14051 IC50 = 133000 nM T33969 C1NC8L 16490 IC50 = 68460 nM T33969 C6RG5E 21233 IC50 = 133000 nM T33969 CJ3OL7 25590 IC50 = 133000 nM T33969 C2N0TD 26070 IC50 = 102700 nM T33969 CJH74G 26596 IC50 > 1000000 nM T33969 CK21BO 27350 IC50 = 133000 nM T33969 CI0W6G 28858 IC50 > 1000000 nM T33969 C68KUD 30627 IC50 > 1000000 nM T33969 C3D2JM 30717 IC50 > 1000000 nM T33969 C4VU9Z 31098 IC50 = 133000 nM T33969 CYP04M 33341 IC50 = 97580 nM T33969 CUJ6W7 35455 IC50 = 73900 nM T33969 CZA2C6 39764 IC50 = 133000 nM T33969 CD9E4R 44668 IC50 > 1000000 nM T33969 CFX82C 47320 IC50 = 133000 nM T33969 CZU9I4 47510 IC50 > 1000000 nM T33969 C6E5CD 48229 IC50 = 133000 nM T33969 CE8LA7 49659 IC50 = 133000 nM T33969 C51MUC 50294 IC50 > 1000000 nM T33969 CU86VK 54459 IC50 = 133000 nM T33969 C7ZUJ4 54840 IC50 = 133000 nM T33969 CC10UB 56801 IC50 = 133000 nM T33969 CQSF39 57004 IC50 = 133000 nM T33969 C4W1LV 58505 IC50 > 1000000 nM T33969 CH8GS0 60749 IC50 = 133000 nM T33969 CYQ4S7 60822 IC50 = 13000 nM T33969 CHZJ65 60834 IC50 = 133000 nM T33969 C2GKD5 62884 IC50 = 133000 nM T33969 CY8ES4 62935 IC50 = 133000 nM T33969 CV4S2E 62969 IC50 = 20500 nM T33969 CA9S6G 62978 IC50 = 45000 nM T33969 C7SO5H 63021 IC50 = 36000 nM T33969 CP8F7B 64143 IC50 = 11800 nM T33969 CD9TC8 64737 IC50 = 133000 nM T33969 C7WUM6 65335 IC50 = 133000 nM T33969 COZ10X 65348 IC50 = 133000 nM T33969 CR23NK 65394 IC50 = 235700 nM T33969 C2E7LR 65493 IC50 = 30000 nM T33969 CS7L6J 65957 IC50 = 133000 nM T33969 C7AV1G 68553 IC50 = 114000 nM T33969 CLAK42 71188 IC50 > 1000000 nM T33969 C73LEV 71399 IC50 = 77000 nM T33969 CYQ3A7 71448 IC50 > 1000000 nM T33969 C6A4VW 71651 IC50 = 133000 nM T33969 CC8U9R 71716 IC50 < 10000 nM T33969 C5UY8O 71950 IC50 > 1000000 nM T33969 CJC4Y8 72067 IC50 = 133000 nM T33969 C2F1OT 77997 IC50 = 133000 nM T33969 C1W8YJ 78000 IC50 = 133000 nM T33969 C6NLX4 84003 IC50 = 133000 nM T33969 CVP7G8 101526 IC50 = 133000 nM T33969 CDY13X 102426 IC50 = 505700 nM T33969 C9T3FB 105007 IC50 < 10000 nM T33969 CPRX31 121899 IC50 = 270600 nM T33969 CIR89V 130211 IC50 > 1000000 nM T33969 C90TYQ 130313 IC50 = 133000 nM T33969 CAR7Y4 146571 IC50 = 133000 nM T33969 CQ3ZD6 150640 IC50 > 892200 nM T33969 C3WVZ6 154068 IC50 = 133000 nM T33969 CPA03B 158789 IC50 > 750900 nM T33969 C3ACD5 161944 IC50 = 111700 nM T33969 C6QWI1 173554 IC50 < 10000 nM T33969 CC3SK9 182176 IC50 > 1000000 nM T33969 CI7BE6 219025 IC50 = 73900 nM T33969 CA6ID2 241903 IC50 = 133000 nM T33969 C8W0LY 249097 IC50 = 31330 nM T33969 CV80FO 249332 IC50 = 133000 nM T33969 C58UBI 253112 IC50 < 10000 nM T33969 C9K1WX 272833 IC50 < 10000 nM T33969 C0VN3D 288216 IC50 = 133000 nM T33969 CLD6J9 441074 IC50 = 133000 nM T33969 CY7HM4 441313 IC50 = 133000 nM T33969 CDU0B1 441351 IC50 = 133000 nM T33969 C82BDA 441371 IC50 = 4100 nM T33969 CDTX86 441405 IC50 < 10000 nM T33969 CVX0K8 443866 IC50 = 133000 nM T33969 C40YBS 444036 IC50 = 133000 nM T33969 C35HJB 656684 IC50 = 22000 nM T33969 C5H4RC 667493 IC50 > 1000000 nM T33969 C8FH0V 667511 IC50 = 133000 nM T33969 CD12VU 667722 IC50 = 13720 nM T33969 CGIY90 688272 IC50 = 133000 nM T33969 CBM17N 3000706 IC50 = 1560 nM T33969 C4BR7C 3005572 IC50 = 115000 nM T33969 CY5ZO7 3032401 IC50 > 1000000 nM T33969 CWQI02 3033817 IC50 = 133000 nM T33969 CH86TV 3033968 IC50 = 133000 nM T33969 C2XP0H 3052775 IC50 = 133000 nM T33969 CX6D4S 3058754 IC50 = 20180 nM T33969 C6TA2Y 3080562 IC50 > 1000000 nM T33969 CL58GA 3085184 IC50 = 606000 nM T33969 CONV41 4022878 IC50 = 133000 nM T33969 C4SL8Q 5281025 IC50 = 133000 nM T33969 C9QDT1 5281067 IC50 = 133000 nM T33969 CNI9X4 5281888 IC50 = 3500 nM T33969 CKTC39 5282139 IC50 > 1000000 nM T33969 C69JBH 5282372 IC50 = 133000 nM T33969 C4X7RJ 5282408 IC50 = 133000 nM T33969 C10CPM 5282455 IC50 = 133000 nM T33969 CBLX43 5282481 IC50 = 133000 nM T33969 CP7B2H 5282593 IC50 > 1000000 nM T33969 CB4P2S 5289394 IC50 = 133000 nM T33969 C0R2YM 5313462 IC50 < 16040 nM T33969 CU6N0T 5351611 IC50 = 164000 nM T33969 CG53MU 5353627 IC50 = 36100 nM T33969 CEP74G 5353634 IC50 = 25590 nM T33969 CUA96S 5388961 IC50 = 133000 nM T33969 CW2C9V 5702125 IC50 = 235600 nM T33969 C5DV8U 5702270 IC50 = 13000 nM T33969 C4GST2 6321416 IC50 = 133000 nM T33969 CC9WJ2 6433334 IC50 = 133000 nM T33969 CO2F7E 6439492 IC50 < 10000 nM T33969 C25BEJ 6440590 IC50 < 10000 nM T33969 CQR03B 6526396 IC50 = 81700 nM T33969 CGM63Y 6540428 IC50 = 33070 nM T33969 C0P8LZ 6602611 IC50 = 87300 nM T33969 CX24OI 6710726 IC50 > 1000000 nM T33969 C1K8VH 6850814 IC50 = 47110 nM T33969 CPK20Z 6917733 IC50 = 133000 nM T33969 C9FQ0W 6918092 IC50 = 133000 nM T33969 CE4TI9 6918427 IC50 = 133000 nM T33969 C1S2RK 6918904 IC50 > 1000000 nM T33969 C9P2HT 9556529 IC50 = 49300 nM T33969 CEO67P 9588170 IC50 = 133000 nM T33969 CE89TG 9799255 IC50 = 39570 nM T33969 C7TMJ6 9799482 IC50 = 18490 nM T33969 C7TN4R 9800927 IC50 = 349200 nM T33969 CE4K0R 9808484 IC50 = 513600 nM T33969 CMIW83 9812710 IC50 < 10000 nM T33969 CEAZ12 9822972 IC50 = 19450 nM T33969 C5W7MS 9833407 IC50 = 133000 nM T33969 CJL94H 9839243 IC50 = 55000 nM T33969 CW86OS 9841004 IC50 > 1000000 nM T33969 C4QFZ6 9841259 IC50 = 105800 nM T33969 C86YFJ 9845843 IC50 < 10000 nM T33969 C9KFV8 9846589 IC50 < 10000 nM T33969 C7QK8R 9847786 IC50 = 133000 nM T33969 C1AW3S 9872994 IC50 < 10000 nM T33969 CDA8I2 9883970 IC50 > 1000000 nM T33969 C7MN9H 9885362 IC50 < 10000 nM T33969 CIWP56 9886273 IC50 = 27700 nM T33969 C5K8NC 9886905 IC50 < 14010 nM T33969 C68EVA 9904199 IC50 < 10000 nM T33969 CMH87T 9905435 IC50 = 22390 nM T33969 C5NH4J 9912089 IC50 = 133000 nM T33969 CGM5Z9 9912499 IC50 < 10000 nM T33969 C7EZN2 9928514 IC50 = 19300 nM T33969 CT0U9F 9929535 IC50 < 10930 nM T33969 C45JHO 9933004 IC50 = 133000 nM T33969 CON68G 9936896 IC50 < 10000 nM T33969 CM28YJ 9949615 IC50 = 49840 nM T33969 CVB57E 10046404 IC50 < 10000 nM T33969 CJK9F8 10046647 IC50 = 124000 nM T33969 C4TL3V 10090208 IC50 < 10000 nM T33969 CIV15Q 10113978 IC50 = 10300 nM T33969 COWN03 10116877 IC50 < 10000 nM T33969 C3T0QX 10119887 IC50 = 55570 nM T33969 CYO93C 10126799 IC50 = 34420 nM T33969 CTAN70 10127634 IC50 < 10000 nM T33969 C37WVJ 10139805 IC50 = 35690 nM T33969 C0NKU8 10183292 IC50 = 22730 nM T33969 CFUO45 10184774 IC50 = 16260 nM T33969 C8T9KD 10194504 IC50 = 19090 nM T33969 CYBM64 10204073 IC50 = 703000 nM T33969 C3FN5E 10226546 IC50 = 247800 nM T33969 C7UPS6 10227020 IC50 < 10000 nM T33969 C9OR4V 10274643 IC50 < 10000 nM T33969 CNPY18 10297363 IC50 = 71540 nM T33969 C5N2US 10310396 IC50 < 10000 nM T33969 C7AY2L 10337564 IC50 < 10000 nM T33969 C5I7MJ 10358698 IC50 < 10000 nM T33969 CZ1XW6 10483360 IC50 = 11500 nM T33969 C8E1UH 10570940 IC50 = 86070 nM T33969 C8BL9W 10695961 IC50 = 133000 nM T33969 CNQK69 10807167 IC50 > 1000000 nM T33969 CGXK13 11176669 IC50 = 106900 nM T33969 C4TK3Q 11294005 IC50 < 10000 nM T33969 CZS5F7 11384286 IC50 < 27030 nM T33969 CV2E4Z 11476710 IC50 = 8530 nM T33969 CU07CF 11556629 IC50 < 13360 nM T33969 CN2T7J 11633897 IC50 = 35840 nM T33969 CA78QO 11677323 IC50 = 32350 nM T33969 CVG4M1 11679357 IC50 = 6490 nM T33969 CL91TM 11968014 IC50 > 1000000 nM T33969 CZ6PB5 12001375 IC50 = 133000 nM T33969 CCLY36 12004215 IC50 = 133000 nM T33969 CYGE17 12358974 IC50 > 1000000 nM T33969 CL2Y7E 13101143 IC50 > 1000000 nM T33969 CO68DY 13543974 IC50 > 1000000 nM T33969 CWI83P 13773524 IC50 < 10000 nM T33969 C78YSK 14091427 IC50 = 364700 nM T33969 C9N5YG 14720269 IC50 = 33900 nM T33969 C42FBS 15765643 IC50 = 14000 nM T33969 CGL5Q2 16051965 IC50 = 133000 nM T33969 CA3JL7 16052011 IC50 = 133000 nM T33969 C7WI4H 16204922 IC50 = 133000 nM T33969 CLHO84 16759173 IC50 = 133000 nM T33969 C71VGO 16760285 IC50 = 133000 nM T33969 CUZE40 18004026 IC50 = 133000 nM T33969 CF8X0D 18422082 IC50 < 10000 nM T33969 C28AYI 18530292 IC50 = 133000 nM T33969 CIVO20 18716149 IC50 > 1000000 nM T33969 C0REQ9 20055509 IC50 = 133000 nM T33969 CH7R8S 20725547 IC50 < 10000 nM T33969 CK6GX1 20725548 IC50 < 10000 nM T33969 CYWQ74 20725549 IC50 < 10000 nM T33969 C3BK5F 21107392 IC50 = 133200 nM T33969 C5CH1W 21337710 IC50 > 135000 nM T33969 CV09WB 21919372 IC50 < 10000 nM T33969 C2Q8OS 21919401 IC50 < 16420 nM T33969 CO32JV 22238181 IC50 < 10000 nM T33969 C93ULY 22718737 IC50 = 55210 nM T33969 C3B2CS 22719722 IC50 < 10000 nM T33969 CQ31BP 23623618 IC50 = 43800 nM T33969 C8JNH4 23666110 IC50 < 11270 nM T33969 CFE9R6 23666879 IC50 = 133000 nM T33969 CH59NC 23667631 IC50 = 133000 nM T33969 C23FRZ 23670523 IC50 > 1000000 nM T33969 CWB0H2 23674512 IC50 = 133000 nM T33969 CFLN18 23675322 IC50 = 133000 nM T33969 CD01LT 23685176 IC50 = 133000 nM T33969 CD53SU 23690471 IC50 < 10000 nM T33969 C9YI0H 23716436 IC50 = 133000 nM T33969 CLJ1S3 24887950 IC50 < 10000 nM T33969 C3N4GQ 25078429 IC50 = 1470 nM T33969 CJ05TN 25210591 IC50 < 10000 nM T33969 CY3CT2 42641861 IC50 = 26810 nM T33969 CW7ZK4 44181971 IC50 = 46000 nM T33969 C1TC4M 45483600 IC50 > 1000000 nM T33969 CUA6N3 46783232 IC50 = 133000 nM T33969 CT6JL8 49799987 IC50 > 969900 nM T33969 C9SCG4 49800073 IC50 = 133000 nM T33969 C0H7OQ 53641749 IC50 > 1000000 nM T33969 CL4G8D 53937048 IC50 < 10000 nM T33969 C1K3LA 54021160 IC50 = 27350 nM T33969 C26TSF 54443266 IC50 < 10000 nM T33969 C5D9TV 54585642 IC50 = 168300 nM T33969 C3RLS2 54677640 IC50 > 1000000 nM T33969 CRV3P5 54685920 IC50 = 133000 nM T33969 CGK7Y9 54685925 IC50 = 133000 nM T33969 CQ6C4E 56972143 IC50 = 15200 nM T33969 C9E8HM 57130306 IC50 = 27550 nM T33969 CM5T1V 57393422 IC50 = 14300 nM T33969 CS7OA6 58516163 IC50 = 10300 nM T33969 CWKF81 59125317 IC50 > 1000000 nM T33969 C1S3LZ 59194184 IC50 = 328700 nM T33969 C76JAL 66577477 IC50 > 983100 nM T33969 CRVI20 67284323 IC50 < 10000 nM T33969 CIMG10 70163838 IC50 = 15890 nM T33969 COVA63 71595704 IC50 = 134900 nM T33969 CI0GU8 71660496 IC50 = 11000 nM T33969 CTO71V 72734347 IC50 = 133000 nM T33969 CRZ62F 73355036 IC50 = 133000 nM T33969 COVK20 90142631 IC50 = 1600 nM T33969 CSM10R 91746235 IC50 > 1000000 nM T33969 C9KV7L 117993993 IC50 = 13300 nM T33969 CMX3U8 118107483 IC50 = 6600 nM T33969 CXD39Z 118170767 IC50 = 4000 nM T33969 C1YK2E 122678192 IC50 = 74000 nM T33969 CZ0O7L 127044281 IC50 = 7000 nM T33969 CF9TC1 131845181 IC50 > 1000000 nM T33969 C41TDB 135413523 IC50 = 132000 nM T33969 CDN1S3 135413539 IC50 = 133000 nM T33969 CG8C4T 135415564 IC50 = 26700 nM T33969 CUN94M 135511839 IC50 > 939800 nM T33969 C5YRP0 135659063 IC50 > 1000000 nM T33969 CKZ45N 137007092 IC50 < 10000 nM T33969 CY1AI4 137007093 IC50 < 10000 nM T33969 C67EFD 137632962 IC50 > 1000000 nM T33969 C84LXT 137642766 IC50 = 65560 nM T33969 C1HB8W 137643646 IC50 > 1000000 nM T33969 C27TMO 137648451 IC50 = 133000 nM T33969 CHPC06 137654606 IC50 = 133000 nM T33969 CJ01GK 137656238 IC50 < 12880 nM T33969 C7F5HY 137658101 IC50 < 10000 nM T33969 C4IH7G 137658562 IC50 < 10000 nM T33969 C0HO6F 137658626 IC50 > 787100 nM T33969 CDU5X4 137658853 IC50 < 10950 nM T33969 C67IKZ 145948937 IC50 = 133000 nM T33969 C2O3LF 145955958 IC50 = 3200 nM T33969 CR9J8V 145957609 IC50 = 1400 nM T33969 CZ8E7J 145959985 IC50 = 300 nM T33969 CMJ50D 145961418 IC50 = 3500 nM T33969 CND38C 155545031 IC50 = 120000 nM T33969 C9RLJ3 3661 IC50 = 133000 nM T33969 D00MFA 134601 IC50 > 1000000 nM T33969 D00REB 11193842 IC50 = 59510 nM T33969 D01BJB 15032 IC50 = 133000 nM T33969 D01OIK 155774 IC50 = 133000 nM T33969 D02YSX 197033 IC50 = 135900 nM T33969 D03IRR 2206 IC50 = 133000 nM T33969 D03IVG 133621 IC50 = 61650 nM T33969 D03ZMQ 323 IC50 > 1000000 nM T33969 D04ALU 3076 IC50 = 82020 nM T33969 D04DLM 2148 IC50 > 1000000 nM T33969 D04LBT 14957 IC50 = 59600 nM T33969 D04SQY 6166 IC50 = 17060 nM T33969 D05BCF 23665591 IC50 = 133000 nM T33969 D05EQG 5265 IC50 < 10000 nM T33969 D05QBF 443375 IC50 < 10000 nM T33969 D05ROV 2757 IC50 > 1000000 nM T33969 D06QBJ 44631903 IC50 = 7000 nM T33969 D07GXY 4850 IC50 = 133000 nM T33969 D07QPA 5280483 IC50 > 1000000 nM T33969 D08CNS 3748 IC50 = 133000 nM T33969 D09NNS 4849 IC50 > 790600 nM T33969 D09XCX 5694 IC50 = 75000 nM T33969 D0F4QX 5601 IC50 = 133000 nM T33969 D0F5LH 4634 IC50 = 27400 nM T33969 D0FO2B 1923 IC50 > 1000000 nM T33969 D0J6JT 1355 IC50 = 133000 nM T33969 D0L9PX 5943 IC50 = 133000 nM T33969 D0M9QJ 44240850 IC50 = 21040 nM T33969 D0O2DQ 237 IC50 = 101100 nM T33969 D0R4PS 135403648 IC50 > 1000000 nM T33969 D0T5RO 16129706 IC50 = 133000 nM T33969 D0V9VJ 4884 IC50 > 1000000 nM T33969 D0Y2JI 5707 IC50 > 1000000 nM T60330 D01BYB 5957 EC50 = 500 nM T60330 D04MSM 2554 IC50 > 100000 nM T60330 D06GDY 43815 IC50 = 1870 nM T60330 D0QL3P 34312 IC50 > 10000 nM T60330 D0UF2N 21706 EC50 = 1000 nM T60330 D08NLQ 114709 IC50 > 100000 nM T60330 C3V0YN 2555 IC50 > 10000 nM T60330 CCP2O5 19099 IC50 > 100000 nM T60330 CXU65D 71013 IC50 > 10000 nM T60330 C67KVL 120031 IC50 > 100000 nM T60330 CPEO63 129274 IC50 = 146000 nM T60330 CV53JZ 135290 IC50 = 72800 nM T60330 C9ZF3M 148882 IC50 = 5970 nM T60330 CT8K5P 179344 IC50 > 20000 nM T60330 CJQ0E1 231766 IC50 > 10000 nM T60330 C50HCD 571066 IC50 = 23300 nM T60330 C0CE1K 606375 IC50 > 100000 nM T60330 CZO07W 738915 IC50 >= 100000 nM T60330 CIWV85 746996 IC50 = 13700 nM T60330 CMUV80 766793 IC50 = 11400 nM T60330 C8DIL6 779112 IC50 >= 100000 nM T60330 CEBX03 779113 IC50 = 34100 nM T60330 CGJ9S2 921624 IC50 = 33800 nM T60330 CYV85L 2320735 IC50 = 420 nM T60330 CI9JA0 2810999 IC50 = 500 nM T60330 C81QCY 2823798 IC50 > 10000 nM T60330 C28EDA 2847675 IC50 > 100000 nM T60330 CA5Z7V 2893185 IC50 = 100000 nM T60330 C6S4CE 3136467 IC50 = 100000 nM T60330 CZ87AQ 3304561 IC50 > 10000 nM T60330 CF2GU9 4281839 IC50 = 100000 nM T60330 CJEV94 5287422 Ki = 48.9 nM T60330 CX92YW 6093160 IC50 > 100000 nM T60330 CA73PI 9841560 IC50 = 350 nM T60330 CQ6NY2 10882078 IC50 = 2490 nM T60330 CX7J8F 11636756 IC50 < 1000 nM T60330 C6LV9U 12231013 IC50 = 26900 nM T60330 CQ81AE 12286268 IC50 > 10000 nM T60330 CC7M9W 12323384 IC50 > 100000 nM T60330 C3I5DQ 12540726 IC50 = 23200 nM T60330 CAB8R9 13644344 IC50 = 4290 nM T60330 CD4S3N 19878631 IC50 > 10000 nM T60330 C98HSJ 20438947 IC50 = 4110 nM T60330 CZF70G 24883277 IC50 > 10000 nM T60330 CG5R0J 40456486 IC50 > 10000 nM T60330 CQ46IG 44353592 EC50 = 490 nM T60330 CWV74N 44579818 IC50 = 10300 nM T60330 CBPD97 46175179 IC50 > 10000 nM T60330 C80DAS 46231312 IC50 > 10000 nM T60330 C2W8ID 46832336 IC50 > 10000 nM T60330 C9ZO8Q 59586810 IC50 > 100000 nM T60330 CO7PZ5 60168729 IC50 = 189 nM T60330 CW9TA8 67474845 IC50 > 100000 nM T60330 CL64YI 70515212 IC50 > 100000 nM T60330 CR2TK8 71324548 IC50 > 10000 nM T60330 CH9Q0R 71450180 IC50 = 2280 nM T60330 C9UC1P 71450181 IC50 = 2640 nM T60330 C4BX9H 71450182 IC50 > 10000 nM T60330 CI2J0Q 71450183 IC50 = 10700 nM T60330 C2YD0P 71452007 IC50 = 52300 nM T60330 C97LUX 71452008 IC50 > 10000 nM T60330 C6KE8N 71452009 IC50 > 10000 nM T60330 C9OI6P 71452010 IC50 > 10000 nM T60330 CFN81R 71453815 IC50 >= 10000 nM T60330 CQO0D5 71453816 IC50 >= 10000 nM T60330 C2Y3CI 71453817 IC50 > 10000 nM T60330 CT0L8R 71455545 IC50 = 3930 nM T60330 C8Y5EX 71455546 IC50 >= 10000 nM T60330 CJN13P 71455547 IC50 = 39100 nM T60330 CX7E4J 71455548 IC50 = 3390 nM T60330 CH5P6D 71455549 IC50 > 10000 nM T60330 CFYW45 71455550 IC50 = 17400 nM T60330 CV9YK5 71457335 IC50 > 10000 nM T60330 CR4D2U 71457336 IC50 > 10000 nM T60330 CR64QG 71457337 IC50 = 1780 nM T60330 CB6Q2R 71457338 IC50 = 12400 nM T60330 CSE07L 71457339 IC50 = 5290 nM T60330 CR1L5W 71459185 IC50 = 2440 nM T60330 C0UOK6 71459186 IC50 > 10000 nM T60330 CJ6F4G 71459187 IC50 >= 10000 nM T60330 C6TI5N 71459188 IC50 = 45800 nM T60330 CSV43Z 71459189 IC50 = 2690 nM T60330 CW87NP 71459190 IC50 > 10000 nM T60330 CA2XU4 71460975 IC50 = 11800 nM T60330 C1LFW8 71460976 IC50 > 10000 nM T60330 C1EXO6 71460977 IC50 = 24600 nM T60330 C0Y1JN 71462707 IC50 = 2350 nM T60330 CPK9Y7 71462708 IC50 = 1020 nM T60330 CK5Z2R 71462709 IC50 = 10800 nM T60330 CWOP84 71462710 IC50 = 9540 nM T60330 C01WEL 71462711 IC50 > 10000 nM T60330 CPE6G0 71657162 IC50 = 54 nM T60330 C3U1YM 73669299 IC50 = 3440 nM T60330 CZPD47 76310105 IC50 >= 100000 nM T60330 CKB8L4 76310106 IC50 > 10000 nM T60330 COJ5W4 76310107 IC50 = 6020 nM T60330 C9C2HW 76313802 IC50 = 52500 nM T60330 C8UA0R 76313803 IC50 = 100000 nM T60330 CX2M6R 76317321 IC50 = 13800 nM T60330 C0G7IA 76317322 IC50 > 20000 nM T60330 CAPZ63 76317323 IC50 = 15300 nM T60330 C43ICX 76317324 IC50 = 27400 nM T60330 C8LY3R 76321046 IC50 >= 100000 nM T60330 C5KG6D 76321047 IC50 >= 100000 nM T60330 C6EXO4 76321048 IC50 > 100000 nM T60330 CEYG95 76321049 IC50 > 100000 nM T60330 CB69EX 76324694 IC50 = 7780 nM T60330 CW1N5Z 76324695 IC50 = 30600 nM T60330 CMZY60 76324696 IC50 = 54600 nM T60330 CF3VQ8 76324697 IC50 = 51400 nM T60330 C5KG2D 76328256 IC50 > 100000 nM T60330 CZL70X 76331932 IC50 >= 100000 nM T60330 CTG6J4 76331933 IC50 > 100000 nM T60330 C8IBW3 76331934 IC50 = 100000 nM T60330 C7QOW9 76331935 IC50 = 19200 nM T60330 C6JW0D 76335511 IC50 = 36200 nM T60330 C69ZBM 76335512 IC50 = 78900 nM T60330 CWP8V1 124125200 IC50 = 84 nM T60330 CPO7N5 124125214 IC50 = 108 nM T60330 CT8V6G 124125228 IC50 = 163 nM T60330 C8IK5C 124125229 IC50 = 8 nM T60330 C2CLF5 124125230 IC50 = 1242 nM T60330 CU79SF 124125231 IC50 = 30 nM T60330 CXKY98 124125238 IC50 = 37 nM T60330 CV05CJ 124125239 IC50 = 10 nM T60330 C0IZ3V 124125244 IC50 = 75 nM T60330 C79JSV 124125246 IC50 = 13 nM T60330 CTY32O 124125268 IC50 = 345 nM T60330 CCZ6E5 124125269 IC50 = 597 nM T60330 CHOK39 124125282 IC50 = 185 nM T60330 CMN43E 124125284 IC50 = 67 nM T60330 CRQI50 124125290 IC50 = 13 nM T60330 CXWS34 124125296 IC50 = 9 nM T60330 CGH4V5 124125301 IC50 = 45 nM T60330 C09UDH 124125305 IC50 = 1681 nM T60330 CGM65Y 124125308 IC50 = 139 nM T60330 CL9JK2 124125309 IC50 = 474 nM T60330 C0HB4J 124125321 IC50 = 134 nM T60330 CSWT23 124125322 IC50 = 93 nM T60330 COTH81 124125330 IC50 = 111 nM T60330 C25LPV 124125335 IC50 = 76 nM T60330 CM2EL8 124125339 IC50 = 88 nM T60330 C2M3UT 124125341 IC50 = 10 nM T60330 CC1B9Y 124125345 IC50 = 317 nM T60330 CT4C9B 124125351 IC50 = 39 nM T60330 C65UQK 124125360 IC50 = 242 nM T60330 C8FN9J 124125383 IC50 = 269 nM T60330 C9J5ZY 124125387 IC50 = 1250 nM T60330 C4SVZ8 124125397 IC50 = 24 nM T60330 C9MI4Q 124125420 IC50 = 2 nM T60330 C84FBW 124125422 IC50 = 173 nM T60330 C0M1TV 124125439 IC50 = 19 nM T60330 CZ92WK 124125444 IC50 = 258 nM T60330 C1PT6B 124125445 IC50 = 5 nM T60330 CL8DB4 124125453 IC50 = 26 nM T60330 C87VMK 124125460 IC50 = 27 nM T60330 C1CDL2 124125463 IC50 = 92 nM T60330 CDJ4H3 124125466 IC50 = 376 nM T60330 C8C7HJ 124125475 IC50 = 52 nM T60330 C2CE8P 124125480 IC50 = 784 nM T60330 CB52JY 124125486 IC50 = 441 nM T60330 CDB27K 124125494 IC50 = 193 nM T60330 C5UJD3 124125495 IC50 = 15 nM T60330 CQ90BD 124125537 IC50 = 2 nM T60330 CZCW68 124125544 IC50 = 2528 nM T60330 CGN86D 124125553 IC50 = 1718 nM T60330 CST92H 136962942 IC50 < 100 nM T60330 CLS0X7 145960885 IC50 > 30000 nM T60330 CWH03B 154731051 IC50 = 260 nM T60330 CF6LV4 155514310 IC50 > 100000 nM T60330 CM9CW2 155526224 IC50 = 12400 nM T60330 C1NOD4 155529242 IC50 = 48000 nM T60330 CX12AU 155529713 IC50 = 11000 nM T60330 C5BC9V 155529971 IC50 > 100000 nM T60330 CMW19R 155530831 IC50 = 430 nM T60330 C1V3EZ 155540682 IC50 > 25000 nM T60330 COD7Q8 155543044 IC50 = 29600 nM T60330 CZ9G8K 155559078 IC50 > 100000 nM T60330 C0PYX1 155562454 IC50 > 30000 nM T60330 D07QYU 4881 EC50 = 10000 nM T60330 D0B0ZQ 9875920 EC50 = 128000 nM T60330 D0B1KT 15953802 IC50 > 10000 nM T60330 D0N6ES 5312126 EC50 = 100000 nM T60330 D0U1OJ 5310983 EC50 = 1000 nM T60330 D0V4GQ 5310996 EC50 = 25000 nM T98155 D0F9FA 5311139 IC50 = 2000 nM T98155 CT7O6B 21580417 IC50 = 4400 nM T98155 C94VLS 57391090 IC50 = 2700 nM T98155 C0P3NW 57398141 IC50 = 15500 nM T98155 CAC6O8 57398142 IC50 = 3700 nM T98155 C5RO1T 57398143 IC50 = 34300 nM T98155 CH41NQ 57401571 IC50 = 37800 nM T98155 CS2UQ8 155535525 IC50 = 7800 nM T17448 CQ9U1Y 16051921 Ki = 19 nM T17448 CTU12O 18008678 Ki = 10400 nM T17448 D09CLP 439155 Ki = 10500 nM T27602 D07XHO 4413 IC50 = 17 nM T27602 D0X9CH 3010818 IC50 > 10000 nM T27602 D05HAD 9955534 Ki = 202000 nM T27602 D0K4FP 44548240 IC50 = 86000 nM T27602 D0Y6SQ 2536 IC50 = 50.6 nM T27602 D02QTV 122267 IC50 = 8 nM T27602 D03QJN 9895762 Ki = 60 nM T27602 D05QMJ 5287596 Ki = 8.1 nM T27602 D08ZCW 9910174 Ki = 66600 nM T27602 D0E2MJ 5496659 Ki = 301 nM T27602 D0G0XN 44342278 Ki = 0.46 nM T27602 D0N7WR 108040 Ki = 290 nM T27602 D0Y5EX 122296 Ki = 0.045 nM T27602 CR8YG3 1308 Ki = 99 nM T27602 C71WRJ 1503 Ki = 6500 nM T27602 CY5B9C 1504 Ki = 6500 nM T27602 C2KE5Q 1508 Ki = 8000 nM T27602 C62ATV 1718 IC50 = 23.7 nM T27602 C72PUR 7504 Ki = 299916251.9 nM T27602 CIF84X 55903 IC50 = 1.6 nM T27602 C0NI8J 55905 IC50 = 27.7 nM T27602 CWO60H 55906 IC50 = 65 nM T27602 CP5XV0 55907 IC50 = 8.4 nM T27602 C4O3YG 55908 IC50 = 18.5 nM T27602 C8DGV7 66035 Ki = 666806769.2 nM T27602 C2HMI7 66036 Ki = 699841996 nM T27602 CRWE01 75452 Ki = 1000000000 nM T27602 C9TN2A 75626 Ki = 8900 nM T27602 CXI6H2 80467 Ki = 3300 nM T27602 CMG15V 122129 Ki = 620 nM T27602 CLX4V7 130395 IC50 = 55 nM T27602 C8AX6L 147654 Ki = 7300 nM T27602 C2WX6R 147797 Ki = 1800 nM T27602 C0TIP9 147804 Ki = 1400 nM T27602 C0M4VW 147922 Ki = 5000 nM T27602 CF95OT 147924 Ki = 293000 nM T27602 CDY9V0 147927 Ki = 9100 nM T27602 CGWP84 147928 Ki = 1100 nM T27602 CQ6VJ0 147929 Ki = 1600 nM T27602 CJ9RY2 147930 Ki = 4300 nM T27602 CLJ6F7 147931 Ki = 8000 nM T27602 CGY1J2 147932 Ki = 10300 nM T27602 C53INQ 147933 Ki = 11100 nM T27602 CZK4S8 147934 Ki = 4800 nM T27602 CDG36W 147935 Ki = 5300 nM T27602 C2U6JH 147936 Ki = 12700 nM T27602 C2JM7B 149831 Ki > 2000000 nM T27602 C1BHS3 193409 Ki = 7780 nM T27602 CZP0Y1 204101 Ki > 10000 nM T27602 C8WZ4I 427814 Ki = 500034535 nM T27602 CU1ZX4 436161 Ki = 357272838.2 nM T27602 CZ17HE 445157 IC50 = 169 nM T27602 C2Z0XW 445482 Ki = 1000 nM T27602 C4W7EG 447219 Ki = 252000 nM T27602 CD0XK3 447221 Ki = 118000 nM T27602 C85OTU 447361 Ki > 2900 nM T27602 CR2DX3 447496 Ki = 1400 nM T27602 COYS31 447502 Ki = 10000 nM T27602 CVI28M 447508 Ki = 320 nM T27602 CS09BE 447510 Ki = 3300 nM T27602 C87OTC 447733 Ki = 2080 nM T27602 CF6D4B 447734 Ki = 56 nM T27602 CHT05K 447735 Ki = 42 nM T27602 C43LRO 448062 Ki = 40 nM T27602 CFMI91 448548 Ki = 150 nM T27602 C5QKC3 448605 Ki = 20 nM T27602 CX5MS1 448610 Ki = 1700 nM T27602 C02CVI 448677 Ki = 23000 nM T27602 CSL82K 449091 Ki = 400 nM T27602 CU3F0X 571728 Ki = 434510224.2 nM T27602 C6HGJ2 2512818 Ki = 399944749.8 nM T27602 CS65PQ 3015798 IC50 = 23.4 nM T27602 CIK93A 3348131 Ki = 30 nM T27602 C69SRC 4292845 Ki = 399944749.8 nM T27602 CFO39X 4369278 Ki = 2100 nM T27602 CPZ6A3 5287506 Ki = 40 nM T27602 C48TEQ 5287836 Ki = 320 nM T27602 C1YGX2 5289320 Ki = 30 nM T27602 C8I0VG 5289529 Ki = 2700 nM T27602 CAW1P7 5497056 Ki = 69 nM T27602 CEB3W0 6426822 Ki = 1000 nM T27602 C2ZRF5 6540265 Ki > 100000 nM T27602 CN57IY 6540268 Ki > 100000 nM T27602 C8OE6S 6913584 IC50 = 11.2 nM T27602 CK64FD 9794516 IC50 = 40 nM T27602 C6JDM9 9799627 Ki = 82 nM T27602 CVFE34 9800775 IC50 > 10000 nM T27602 C2FHU7 9801905 IC50 = 23 nM T27602 CL1R0T 9801948 Ki > 100000 nM T27602 C40LRN 9802229 Ki = 2900 nM T27602 CYL75R 9802758 Ki = 6800 nM T27602 C3FS0U 9802858 Ki = 10000 nM T27602 C4VX9Y 9803558 IC50 > 10000 nM T27602 C07DSH 9804052 Ki = 1600 nM T27602 C8QGS1 9804434 Ki > 1500 nM T27602 C1FIN6 9804775 IC50 > 130 nM T27602 C4OTK6 9805415 IC50 > 10000 nM T27602 CAKN38 9805632 Ki > 1600 nM T27602 C6JIT7 9806444 IC50 > 11000 nM T27602 CBKL18 9806644 IC50 = 9820 nM T27602 CAG59M 9808035 Ki = 850 nM T27602 C8UX0O 9810198 Ki = 34000 nM T27602 CKN89B 9822176 Ki = 860 nM T27602 CD5M9P 9823195 Ki = 100000 nM T27602 CJ2G7A 9823668 IC50 = 3370 nM T27602 CD3AP6 9824122 Ki > 1500 nM T27602 C0QH1L 9824657 Ki = 213000 nM T27602 CZ64PW 9824925 Ki > 1500 nM T27602 C08XFQ 9825841 Ki = 49.3 nM T27602 CPB20R 9826345 Ki = 1200 nM T27602 CS1DL7 9826716 IC50 = 970 nM T27602 CB82VS 9827306 IC50 > 11000 nM T27602 CE0HD3 9828470 Ki = 19900 nM T27602 COW7Q3 9829120 IC50 = 2400 nM T27602 C4F8CN 9830285 IC50 = 420 nM T27602 CGNB60 9830581 IC50 = 2100 nM T27602 C6W8QC 9831694 IC50 = 378000 nM T27602 C1WK3X 9838954 Ki = 77000 nM T27602 C58QBT 9842536 Ki > 15000 nM T27602 C14HZE 9842688 Ki > 1000000 nM T27602 CVO5R3 9842851 IC50 > 10000 nM T27602 C7UOA2 9844807 Ki = 120000 nM T27602 CC4Y8V 9845104 Ki = 4500 nM T27602 CY7FU4 9846410 Ki = 6100 nM T27602 C8I4LS 9846496 Ki > 1500 nM T27602 C5Z2RH 9848091 IC50 > 11000 nM T27602 CW3EC6 9848592 Ki = 210 nM T27602 CCL5G3 9848846 IC50 = 1250 nM T27602 CY7B8Q 9860803 Ki = 233000 nM T27602 CF74PR 9864759 IC50 > 10000 nM T27602 CSH3K5 9865994 Ki = 4300 nM T27602 CY6EA8 9868194 Ki = 6300 nM T27602 CL6QS0 9868922 Ki = 3.3 nM T27602 CZ9LR2 9870910 Ki = 1100 nM T27602 CIL85V 9871029 IC50 > 11000 nM T27602 C9UB6X 9871197 Ki > 1500 nM T27602 CIZ61P 9872423 Ki > 68300 nM T27602 C6ZB3K 9872552 IC50 > 11000 nM T27602 C87SWZ 9872983 Ki = 84000 nM T27602 CG0L6A 9873029 IC50 = 4000 nM T27602 CJ1XE3 9874681 IC50 = 9700 nM T27602 CA9Z4S 9875345 Ki = 39000 nM T27602 CJT9X7 9887558 Ki = 282 nM T27602 CAW39H 9888145 Ki = 290000 nM T27602 CL61HY 9888442 IC50 > 100000 nM T27602 CG2EZ0 9889108 IC50 < 100000 nM T27602 CYKX52 9889871 Ki = 740 nM T27602 C6A4TL 9890540 Ki > 1500 nM T27602 C17NPU 9890541 IC50 = 26.2 nM T27602 CO4KT2 9891302 Ki = 810 nM T27602 CD13TH 9891795 IC50 > 10000 nM T27602 C1M2PU 9892103 IC50 > 11000 nM T27602 CXY68Z 9893122 IC50 = 5170 nM T27602 C5T0GJ 9895523 IC50 = 490 nM T27602 C6PSQ7 9896889 Ki = 15000 nM T27602 C0SP6Q 9906596 Ki = 320 nM T27602 C2HN7L 9907201 Ki = 110 nM T27602 C85SEZ 9908687 IC50 > 10000 nM T27602 C7KJP3 9908917 IC50 > 100000 nM T27602 CQ7PT5 9910790 Ki = 1100 nM T27602 C5HS9Y 9911866 Ki = 3200 nM T27602 C21RUG 9911960 Ki = 61000 nM T27602 CL0K6H 9912101 Ki = 1600 nM T27602 CS6QF5 9912191 Ki > 1500 nM T27602 C8GJF3 9913055 IC50 = 101 nM T27602 C1C3VT 9914538 IC50 > 11000 nM T27602 CC0D5H 9915041 Ki = 3500 nM T27602 CK2H1C 9917705 Ki = 45 nM T27602 CFO1K9 9922130 Ki = 7000 nM T27602 CLZ53G 9922131 Ki = 6900 nM T27602 CAP64B 9929157 Ki = 96 nM T27602 C7ZJ5X 9931673 Ki > 100000 nM T27602 CS7LF5 9931725 Ki = 2000 nM T27602 CRD3A7 9931726 Ki > 100000 nM T27602 C9I2ES 9931785 IC50 = 560 nM T27602 CGT3K4 9932145 IC50 > 100000 nM T27602 CG3B1P 9935390 Ki = 600 nM T27602 CL2NV0 9935925 IC50 = 360 nM T27602 C5KS0R 9936020 IC50 > 11000 nM T27602 CKLJ26 9936190 IC50 = 64 nM T27602 C49DRC 9936691 IC50 > 11000 nM T27602 CL0U1E 9936850 IC50 = 189 nM T27602 CG96QC 9936983 Ki = 98 nM T27602 COA4R0 9937032 Ki = 170 nM T27602 C8F5CW 9937921 Ki = 60 nM T27602 C1RHT8 9949886 Ki = 130 nM T27602 CD27EJ 9951054 IC50 = 2700 nM T27602 COR74I 9954289 Ki = 431000 nM T27602 CWNA41 9954607 Ki = 1000 nM T27602 C0R4GE 9954812 IC50 = 1200 nM T27602 CP7A2W 9955292 Ki > 1500 nM T27602 CSI62L 9955475 IC50 > 10000 nM T27602 C3EPC4 9955758 Ki > 22000 nM T27602 CV96ZD 9955999 Ki > 1500 nM T27602 CM7IF6 9956559 Ki = 570 nM T27602 C8CLF7 9956947 Ki = 1400 nM T27602 CI84CP 9957386 Ki > 5200 nM T27602 CE39JM 9958168 Ki = 140 nM T27602 C3WAS5 9958320 Ki = 2200 nM T27602 C9AW3Q 9958913 IC50 < 1 nM T27602 C2Y0QV 9959268 IC50 > 10000 nM T27602 CBC2K3 9959749 IC50 > 11000 nM T27602 C0C1FQ 9959919 Ki > 4200 nM T27602 C2CE1A 9962331 Ki > 50000 nM T27602 C0TV8Q 9962561 Ki = 153000 nM T27602 C5SA7F 9983043 IC50 = 135 nM T27602 CZ3U8E 9984568 Ki = 48000 nM T27602 CU9QI6 10004529 Ki = 6.4 nM T27602 C8I7YZ 10006319 IC50 = 17 nM T27602 CFQV59 10007890 IC50 > 10000 nM T27602 CWMC62 10009177 IC50 = 590 nM T27602 C98OVC 10021822 Ki = 77000 nM T27602 CDF1Q4 10025885 Ki = 860 nM T27602 CBL8D4 10026170 Ki = 2.5 nM T27602 CF1V4K 10027758 Ki > 2900 nM T27602 CW5JH1 10028252 Ki = 80 nM T27602 CX4TI5 10029172 Ki = 64 nM T27602 C3E4DR 10029213 IC50 = 24 nM T27602 CI2O5B 10029343 IC50 > 11000 nM T27602 C8KIA9 10037020 IC50 = 0.12 nM T27602 C08PUS 10051441 IC50 = 13 nM T27602 C29DTM 10051582 Ki = 150 nM T27602 CU9I7D 10051599 Ki = 52 nM T27602 CHZL08 10051960 Ki = 70 nM T27602 CFCT67 10053115 Ki = 3800 nM T27602 CBV7N2 10070407 IC50 = 19 nM T27602 CPR1C7 10070588 Ki = 140000 nM T27602 C2RNL5 10071434 IC50 > 100000 nM T27602 CB04YW 10073864 IC50 = 32 nM T27602 CF4R2W 10074230 IC50 = 9.8 nM T27602 C9ZCS2 10074922 IC50 = 19 nM T27602 CD5AT6 10075317 Ki = 5000 nM T27602 C2CUX3 10075442 Ki = 93 nM T27602 CR0ZL7 10091675 IC50 = 19 nM T27602 C1HIC3 10093417 Ki = 200000 nM T27602 CEN06H 10093642 IC50 = 4.13 nM T27602 C3TDM1 10094168 Ki = 69 nM T27602 C2VT9U 10094219 Ki = 76 nM T27602 C3TWI1 10095455 Ki > 100000 nM T27602 CW6LB3 10097039 Ki = 1850 nM T27602 CQB1V2 10101474 IC50 = 0.2 ug.mL-1 T27602 CMOE48 10113121 Ki = 4.4 nM T27602 C0AFU1 10116445 Ki > 2900 nM T27602 CW4RZ5 10116936 IC50 > 450 nM T27602 CXCR46 10117543 Ki > 68000 nM T27602 CV5E4L 10121049 Ki > 68300 nM T27602 CR03NV 10131788 Ki = 14000 nM T27602 CVA35H 10140425 Ki > 168 nM T27602 CS2G4T 10140847 Ki = 3.5 nM T27602 CMFW67 10140911 Ki > 2500 nM T27602 CWF4I3 10141502 Ki = 67000 nM T27602 C7L5IJ 10157296 Ki = 45 nM T27602 C4K3WG 10162441 Ki = 13.6 nM T27602 CT65YJ 10162799 Ki = 110 nM T27602 CBHY78 10163266 Ki = 31.3 nM T27602 CF82TK 10163421 Ki > 5200 nM T27602 C75ADN 10164065 Ki > 5200 nM T27602 CM6PS4 10165173 Ki = 47000 nM T27602 C5WB4J 10165649 Ki > 68300 nM T27602 C7G4JC 10166616 Ki > 68300 nM T27602 CEPJ05 10166622 Ki > 68300 nM T27602 CT31ZH 10183608 Ki = 18.7 nM T27602 C7PC2K 10185292 IC50 > 170 nM T27602 C93EKT 10185327 Ki = 11.9 nM T27602 C1DN4F 10187311 Ki = 216600 nM T27602 CHY62J 10203373 Ki > 1600 nM T27602 C01QTR 10209142 Ki > 68300 nM T27602 C8V1AY 10225952 Ki = 11 nM T27602 C6HAC0 10227428 Ki > 1600 nM T27602 CT18AE 10227443 Ki > 2900 nM T27602 CIAX57 10228506 Ki = 32000 nM T27602 C98FSX 10230007 Ki = 17000 nM T27602 C2XHG8 10248900 Ki = 880 nM T27602 C9QML3 10250104 Ki = 760 nM T27602 C7RVY1 10253674 Ki = 1260 nM T27602 C4Z1LU 10255253 Ki > 2900 nM T27602 C4WV1A 10257345 IC50 = 169 nM T27602 C9E8OU 10273521 Ki = 19.7 nM T27602 C0J1TD 10278414 Ki = 40 nM T27602 C3M5KS 10279315 Ki = 415 nM T27602 CB1S5P 10281431 Ki > 68300 nM T27602 CZM97W 10293977 Ki = 3400 nM T27602 C5EDW1 10294146 Ki = 30 nM T27602 CEW97F 10301102 Ki = 53 nM T27602 C8XLH9 10302418 Ki = 415800 nM T27602 CGTF74 10303947 Ki > 68300 nM T27602 C8PA9J 10310498 Ki > 1600 nM T27602 CMR6Y8 10323469 IC50 = 9700 nM T27602 C41ZLB 10326602 IC50 = 97.8 nM T27602 CH0X3M 10337666 IC50 > 100000 nM T27602 CP64HV 10342843 Ki = 350 nM T27602 CFL57Y 10343633 Ki = 150 nM T27602 C9XUD8 10347489 IC50 = 440 nM T27602 C4KER5 10347610 IC50 = 4390 nM T27602 CK87NT 10348221 Ki = 4000 nM T27602 CHC08V 10349473 IC50 = 11000 nM T27602 CH0V8B 10366070 Ki = 560 nM T27602 C10ISY 10367012 Ki = 120 nM T27602 C1D4YB 10367245 Ki = 1930 nM T27602 CJ0O5P 10367277 IC50 = 935 nM T27602 CG98CM 10367552 Ki = 63 nM T27602 CJWE07 10368488 IC50 = 13 nM T27602 CDO83F 10368538 Ki = 13000 nM T27602 C26CSM 10386393 IC50 = 18 nM T27602 CG2WB8 10387708 Ki = 0.24 nM T27602 C7TH5Q 10387956 Ki > 1600 nM T27602 CMNP39 10389039 IC50 > 10000 nM T27602 CSC52L 10390341 IC50 = 1900 nM T27602 CJNV62 10391699 IC50 = 10005 nM T27602 CLK08Z 10391999 IC50 > 10000 nM T27602 CM1WJ6 10394292 Ki = 120 nM T27602 CCL85B 10394816 IC50 = 300 nM T27602 C56NXW 10409551 IC50 = 570 nM T27602 C03MWI 10413130 Ki = 540 nM T27602 CJTH60 10432907 Ki = 11 nM T27602 C1RE8V 10433463 IC50 = 174 nM T27602 CX39AB 10435238 Ki = 420 nM T27602 C48HDV 10435701 Ki = 9300 nM T27602 C9K5GO 10436126 Ki = 37000 nM T27602 CUM2T7 10436294 Ki = 45 nM T27602 CG07WY 10438196 Ki = 47 nM T27602 C9HI6A 10460541 IC50 = 1.5 nM T27602 CI87FD 10460564 IC50 = 31 nM T27602 CWG91R 10472893 Ki = 930 nM T27602 C45KWI 10480373 Ki = 140 nM T27602 CCP2N8 10480374 Ki > 2900 nM T27602 CV0X6G 10480463 IC50 > 11000 nM T27602 CM5A3J 10481558 Ki = 5 nM T27602 CMIN26 10481978 Ki = 120 nM T27602 CG18KR 10483116 Ki = 25180 nM T27602 CJ50AY 10483408 Ki = 80 nM T27602 CY16UR 10504366 Ki = 610 nM T27602 CXB50R 10508061 Ki = 260 nM T27602 C87BCM 10525391 Ki = 820 nM T27602 C42XPE 10526785 Ki = 300 nM T27602 CU8I0J 10528552 Ki = 160 nM T27602 C5ED3G 10529121 Ki = 18000 nM T27602 C1K0NS 10532026 Ki = 300 nM T27602 CKYZ01 10532259 Ki = 100 nM T27602 CK13IY 10546004 Ki = 870 nM T27602 C37BYS 10548542 Ki = 1200 nM T27602 CCM1I8 10552861 Ki = 17000 nM T27602 CYX1V7 10553919 Ki = 221 nM T27602 CE8V0B 10555065 Ki = 470 nM T27602 CQG10I 10556031 Ki = 67 nM T27602 CSK8V5 10556085 Ki = 330 nM T27602 CGHL47 10556206 Ki = 120 nM T27602 CY1JF2 10569959 Ki = 820 nM T27602 C52FQT 10571832 Ki = 140 nM T27602 C6LO8Q 10580222 Ki = 120 nM T27602 C1D8GI 10580396 Ki = 110 nM T27602 C42LVU 10580437 Ki = 72 nM T27602 C02RYN 10592155 Ki = 1200 nM T27602 C4VMO3 10595198 Ki = 330 nM T27602 C8P3QI 10599262 Ki = 2100 nM T27602 CCQU28 10600245 Ki = 270 nM T27602 CP69LR 10604270 Ki = 340 nM T27602 CY1J0N 10604774 Ki = 49 nM T27602 C8ZXS3 10609754 IC50 = 0.02 nM T27602 C1RH3P 10621200 Ki = 110 nM T27602 CO83BP 10622800 IC50 = 1200 nM T27602 CV0I5Y 10623890 Ki = 600 nM T27602 C03CIN 10628066 Ki = 350 nM T27602 C4M0QB 10645022 Ki = 220 nM T27602 CFNH06 10645807 IC50 = 990 nM T27602 CR1Y2D 10647704 Ki = 340 nM T27602 C6E4WZ 10651873 Ki = 54 nM T27602 CBT96N 10664145 Ki = 1400000 nM T27602 CJG9H6 10669349 Ki = 29000 nM T27602 C7CVW2 10669933 IC50 = 1100 nM T27602 CIKJ09 10672223 Ki = 390 nM T27602 CP6RF7 10673965 IC50 = 118 nM T27602 CM1Y2D 10675086 Ki = 310 nM T27602 C8P2UC 10675884 Ki = 300 nM T27602 CJPN01 10694782 Ki = 94 nM T27602 CIB63V 10694800 Ki = 41 nM T27602 CW8RV0 10696389 Ki = 180 nM T27602 CP4QC5 10696511 Ki = 1600 nM T27602 C3QH0L 10697320 Ki = 98 nM T27602 CY0P5F 10714145 Ki = 480 nM T27602 CF6TZ2 10715258 Ki = 440 nM T27602 CCP58N 10718840 Ki = 120 nM T27602 CIKF89 10719580 Ki = 2500 nM T27602 CAS17I 10722747 Ki = 25 nM T27602 CUTA38 10723163 Ki = 49 nM T27602 CZ0Q8K 10742217 Ki = 9000 nM T27602 C7RWD8 10744643 Ki = 27000 nM T27602 C5DYQ3 10769476 Ki = 250 nM T27602 C62KFB 10769759 Ki = 41 nM T27602 C5E6AY 10770527 Ki = 90 nM T27602 C4Z2LQ 10770606 Ki = 47 nM T27602 CQW74C 10770621 Ki = 91 nM T27602 CCZ9U0 10770773 Ki = 200 nM T27602 C3W7TF 10770845 Ki = 72 nM T27602 C5ENU2 10794450 Ki = 18 nM T27602 C64ZVF 10794532 Ki = 120 nM T27602 CC95IV 10794535 Ki = 80 nM T27602 CD6U1P 10806942 Ki > 1200 nM T27602 C3WX4F 10813359 Ki = 47 nM T27602 CSZR21 10817699 Ki = 390 nM T27602 CUS6D0 10818009 Ki = 180 nM T27602 C2D1KY 10820951 IC50 = 41 nM T27602 C9HPZ8 10831834 IC50 = 4300 nM T27602 CJ0KB8 10835917 Ki = 4800 nM T27602 CM13CR 10840852 Ki = 240 nM T27602 CYX51H 10840933 Ki = 83 nM T27602 C2R7OQ 10841758 Ki = 70 nM T27602 CBK06L 10861643 IC50 > 100000 nM T27602 CKG30N 10863633 Ki = 567000 nM T27602 CN6WO8 10863757 Ki = 720 nM T27602 C48IUK 10864508 Ki = 9.1 nM T27602 CXG62W 10874449 Ki > 2900 nM T27602 C2TH3I 10875009 Ki > 2900 nM T27602 CN74ZX 10884041 Ki = 3800 nM T27602 C19DGJ 10884304 Ki = 1600 nM T27602 C30EGA 10885646 Ki = 260 nM T27602 C2MV8C 10886082 Ki = 4 nM T27602 C1VRY3 10895218 Ki = 270000 nM T27602 CQTC02 10903566 Ki = 1600 nM T27602 C8J1TX 10904089 Ki = 23000 nM T27602 CUMI91 10905246 Ki > 100000 nM T27602 C7E3AJ 10906300 Ki = 1400 nM T27602 CH2G5Q 10906977 Ki > 68000 nM T27602 CK68OT 10927655 Ki = 4600 nM T27602 C5KM8X 10928726 Ki = 370 nM T27602 CDWG32 10938987 Ki = 800 nM T27602 C8OA1L 10946869 Ki = 17000 nM T27602 CITU70 10962439 Ki > 68000 nM T27602 CS1AL4 10983261 Ki = 2900 nM T27602 C6ST2N 10983389 Ki = 9200 nM T27602 CQGL23 10983472 Ki = 706000 nM T27602 CL9V7T 10984300 Ki > 2900 nM T27602 C8NHR5 10984568 Ki = 7 nM T27602 CVI57D 10994262 Ki = 700 nM T27602 CUV8Q3 11004075 Ki = 3600 nM T27602 C43SNO 11004109 Ki = 1000 nM T27602 C7FP6L 11004280 Ki > 1000000 nM T27602 C7JQ3S 11005330 Ki = 550 nM T27602 C8L2WC 11005945 Ki = 53 nM T27602 CC39SB 11009950 Ki = 55000 nM T27602 CYZL25 11015002 Ki = 700 nM T27602 C69FOW 11025238 Ki = 898000 nM T27602 C4IE3S 11026399 Ki = 501000 nM T27602 C4ZPT7 11037871 Ki = 7900 nM T27602 CYNU74 11048541 Ki = 40000 nM T27602 CPEK84 11048789 Ki = 89 nM T27602 C4SW1T 11049045 Ki > 2900 nM T27602 CD9WJ8 11057540 Ki = 130 nM T27602 C2Y6VW 11057779 Ki = 75 nM T27602 CH1OX5 11059588 Ki > 2900 nM T27602 C8BC4U 11059598 Ki > 2900 nM T27602 C3HNB2 11068806 Ki = 4300 nM T27602 C8ELX0 11070538 Ki = 7300 nM T27602 CP4R1J 11070822 Ki = 1100 nM T27602 C29EIG 11079364 Ki = 251000 nM T27602 CSE89U 11081058 Ki > 2900 nM T27602 CV0AS6 11091843 Ki = 665000 nM T27602 CAW0O5 11092493 IC50 = 240 nM T27602 CKL74M 11113517 Ki > 2900 nM T27602 C4K6YA 11123202 Ki = 429000 nM T27602 CEG83K 11135464 Ki = 9.9 nM T27602 C9KL8Y 11144992 Ki > 2900 nM T27602 CAD15G 11149953 Ki = 2610 nM T27602 C3WKQ1 11168297 Ki > 1500 nM T27602 CEK78H 11181141 Ki = 300 nM T27602 C6LVG4 11186243 Ki = 260 nM T27602 CTX9F3 11188793 Ki = 115 nM T27602 CJ6CW4 11203935 Ki > 2500 nM T27602 C8BRJ1 11225386 Ki > 1500 nM T27602 CP51FI 11226542 Ki > 1600 nM T27602 CHLK70 11244460 Ki = 235 nM T27602 C98HOZ 11249318 Ki > 1600 nM T27602 C86DZB 11292119 Ki = 43 nM T27602 C0TUI9 11307532 Ki > 1600 nM T27602 CVAI21 11330048 Ki > 2500 nM T27602 C64EOX 11341794 Ki > 2500 nM T27602 C6CDN3 11347670 Ki = 1320 nM T27602 CLY5G8 11350400 Ki = 58 nM T27602 CG85IF 11356901 Ki = 29991625.19 nM T27602 CTJ1Z2 11361949 Ki = 39 nM T27602 C8URO7 11387451 Ki > 1600 nM T27602 CODR29 11420832 Ki = 18000 nM T27602 CM7DK5 11445304 Ki > 1600 nM T27602 C8KJ1G 11466928 Ki > 2500 nM T27602 CH4V9C 11468062 Ki > 4200 nM T27602 C63LIR 11473486 Ki = 51 nM T27602 CU04WZ 11478333 Ki > 1600 nM T27602 CVI82D 11479420 Ki > 5200 nM T27602 CS12RM 11730232 Ki > 2900 nM T27602 CQ0ZP6 11730472 Ki > 2900 nM T27602 CN6X4B 11733626 Ki = 136000 nM T27602 CQ5U8H 11739438 Ki = 92 nM T27602 CM95SZ 11744578 IC50 = 259 nM T27602 CNPW05 11755188 IC50 > 10000 nM T27602 CUMO51 11756555 IC50 > 10000 nM T27602 CS0JR2 11756961 Ki = 17 nM T27602 C83GXL 11757017 IC50 = 4000 nM T27602 C07WYX 11762017 Ki = 855 nM T27602 C4F0HE 11762405 Ki = 80000 nM T27602 CZ91LI 11762766 Ki > 68000 nM T27602 C7JLR1 11774107 Ki = 13 nM T27602 CR2E9T 11782463 Ki = 290 nM T27602 CMH70L 11784384 Ki = 1600 nM T27602 CP2I9G 11796404 Ki = 1500 nM T27602 C8EHN3 11797101 Ki = 2600 nM T27602 CH2Z1N 11798267 Ki = 1500 nM T27602 C68VNG 11801427 Ki = 390 nM T27602 CL01GT 11801580 Ki = 120 nM T27602 CVZ82O 11801725 Ki = 390 nM T27602 CFP36D 11802531 Ki = 113 nM T27602 CY46UZ 11802721 Ki = 290 nM T27602 CO5X8E 11811735 Ki > 1000000 nM T27602 CL0W8P 11812192 Ki = 5000 nM T27602 CPR54N 11812296 Ki = 800 nM T27602 CZIB40 11812370 Ki = 47000 nM T27602 C4XE8C 11812643 Ki = 1600 nM T27602 C9VW2P 11813305 Ki > 2900 nM T27602 C98ZOR 11824040 Ki = 1200 nM T27602 CIO26S 11826929 Ki = 5000 nM T27602 C6UT2G 12042266 Ki = 4200 nM T27602 CQG4D9 12042267 Ki = 510 nM T27602 CBL13C 12042268 Ki = 22000 nM T27602 C7OC2I 12042269 Ki = 12700 nM T27602 CPR4I1 12047383 Ki = 1320 nM T27602 C5U0FJ 12047384 Ki = 1780 nM T27602 C5FU3H 12047385 Ki = 126000 nM T27602 CZ9S6D 12314068 Ki = 2300 nM T27602 C4MTL2 12925726 IC50 = 17.2 nM T27602 C7PNY5 12925730 IC50 = 19 nM T27602 CW4EJ0 12925742 IC50 = 16.5 nM T27602 CPB09W 13192674 IC50 = 45900 nM T27602 CO0J3T 13192685 IC50 = 163800 nM T27602 CO2LB0 13236162 Ki = 1800 nM T27602 C4LF8R 13236165 Ki = 3800 nM T27602 CB0I7H 13236166 Ki = 4000 nM T27602 CTH7S1 13245173 Ki = 2700 nM T27602 C4SJ8H 13245401 IC50 = 1.5 nM T27602 CDG80P 13245402 IC50 = 300 nM T27602 CV9UK1 13590035 IC50 = 27.1 nM T27602 C0IH5M 13712401 IC50 = 12.6 ug.mL-1 T27602 C2DGN3 14046022 IC50 = 1500 nM T27602 CA26FM 14480651 IC50 = 87.6 nM T27602 CIB7M6 14480685 IC50 = 92.2 nM T27602 CY87AI 14488960 IC50 = 107100 nM T27602 CM8W7C 14488962 IC50 = 81400 nM T27602 C6VM2S 14488964 IC50 = 195700 nM T27602 CK5Z7P 14488966 IC50 = 400000 nM T27602 C7EIL0 14488968 IC50 = 400000 nM T27602 C50XDQ 14488970 IC50 = 400000 nM T27602 C54JLM 14488972 IC50 = 400000 nM T27602 C0WSE1 14488974 IC50 = 400000 nM T27602 CH9I4M 14488976 IC50 = 400000 nM T27602 C5CK1E 14488978 IC50 = 400000 nM T27602 C0M1PW 14645136 Ki = 1500 nM T27602 CC09SA 14645140 Ki = 1300 nM T27602 C06BKJ 14645142 Ki = 1300 nM T27602 C8MH7S 14645147 Ki = 1100 nM T27602 C67ZIM 14645153 Ki = 5400 nM T27602 CJ6S1W 14645154 Ki = 1000 nM T27602 CIE47P 15434242 Ki = 1900 nM T27602 CZBD56 15435386 Ki = 480 nM T27602 CY42MO 15449319 IC50 = 0.6 nM T27602 CFJB64 15449320 IC50 = 2 nM T27602 C48WFU 15449321 IC50 = 26 nM T27602 CGX57Z 15454127 Ki = 101000 nM T27602 CKH1S3 15458385 Ki = 550 nM T27602 C5CQ6R 15463576 Ki = 52 nM T27602 CCN18Q 15463577 Ki = 200 nM T27602 CY2S1U 15463580 Ki = 110 nM T27602 CQTF26 15463581 Ki = 750 nM T27602 CX5S1Z 15511974 Ki = 160 nM T27602 CKGJ08 15516769 IC50 = 340 nM T27602 C5Z4MG 15516770 IC50 = 9100 nM T27602 CP63GF 15534822 IC50 = 289 nM T27602 C5NQH0 15541215 IC50 = 1300 nM T27602 CL4DX2 15541216 IC50 = 5830 nM T27602 CP7ZC9 15541217 IC50 = 1500 nM T27602 CQ09TY 15541218 IC50 = 930 nM T27602 CQ20FX 15541219 IC50 = 4500 nM T27602 CRV96C 15541220 IC50 > 100000 nM T27602 CWX23I 15541221 IC50 = 10100 nM T27602 CC43YL 15541222 IC50 = 8300 nM T27602 C2BZ4F 15541223 IC50 > 100000 nM T27602 CJ8U1I 15541224 IC50 > 100000 nM T27602 C65BNG 15541225 IC50 > 200000 nM T27602 C4XDQ6 15541226 IC50 = 4200 nM T27602 CWM38R 15541227 IC50 = 2200 nM T27602 CPJT95 15545832 Ki > 2900 nM T27602 CP3DF2 16776143 Ki = 199986187 nM T27602 CT6EN9 16794642 Ki = 299916251.9 nM T27602 CTQ85L 18397340 Ki = 28000 nM T27602 CZ4L5C 18397341 Ki = 445000 nM T27602 CU5N8E 18397342 Ki = 850000 nM T27602 C4HE7G 18397344 Ki = 66000 nM T27602 CF1Y7P 18397345 Ki = 171000 nM T27602 C3D1VS 18397346 Ki = 21000 nM T27602 CEJ3K1 18397347 Ki > 1000000 nM T27602 CVB47A 18397350 Ki > 1000000 nM T27602 C7DB0W 18397352 Ki = 25000 nM T27602 C03OYT 18397353 Ki > 1000000 nM T27602 CP3ZL0 18397354 Ki = 219000 nM T27602 CM28UY 18397357 Ki = 82000 nM T27602 C0POA1 18397359 Ki = 754000 nM T27602 CSW0L3 18397360 Ki > 1000000 nM T27602 CN9S6X 18397370 Ki = 129000 nM T27602 CS21RN 18397380 Ki > 1000000 nM T27602 C9NB0Z 18675062 IC50 = 300 nM T27602 C09KIY 18675079 IC50 = 760 nM T27602 C29WYS 18675086 IC50 = 330 nM T27602 CR6I5L 18675103 IC50 = 39000 nM T27602 CLZ97R 18675188 IC50 = 13000 nM T27602 CK6U1I 18675238 IC50 = 2500 nM T27602 CN0LW2 18675252 IC50 = 7800 nM T27602 CD9UE4 18675298 IC50 = 2100 nM T27602 CB0IQ4 18727607 IC50 > 11000 nM T27602 C31ZAL 18727831 IC50 > 11000 nM T27602 CJY67O 18727833 IC50 > 11000 nM T27602 C02HEA 18727834 IC50 > 11000 nM T27602 CJSL38 18727836 IC50 > 11000 nM T27602 C8AMY9 18727838 IC50 > 11000 nM T27602 CY8AC3 18727841 IC50 > 11000 nM T27602 CD02TK 18727852 IC50 > 11000 nM T27602 C1JMX5 18727855 IC50 > 11000 nM T27602 CNUR53 18800583 Ki = 130 nM T27602 CMA2G0 18800591 Ki > 15000 nM T27602 CX46SV 20113118 Ki = 399944749.8 nM T27602 CY2IO0 20115763 Ki = 100000000 nM T27602 CO2JG4 20595081 IC50 > 11000 nM T27602 CM7BH1 20595091 IC50 > 11000 nM T27602 CCH5N1 20595225 IC50 > 11000 nM T27602 C2ID8R 20595260 IC50 > 10000 nM T27602 CMT46A 20595328 IC50 > 10000 nM T27602 C7LHE8 20641745 IC50 = 39.1 nM T27602 CTY8G2 20707887 Ki = 36 nM T27602 CS3HB4 20801160 Ki > 100000 nM T27602 CR6C2I 21218691 Ki = 700 nM T27602 CS5L2M 21218709 Ki > 1200 nM T27602 CEQ6B2 21218732 Ki = 630 nM T27602 C79ZNM 21218751 Ki > 1200 nM T27602 CGC48U 21250249 IC50 = 3500 nM T27602 CNTI15 21366511 IC50 > 11000 nM T27602 C5S8ZW 21366513 IC50 > 11000 nM T27602 C67QCO 21366574 IC50 > 11000 nM T27602 CS2L1Y 21366575 IC50 > 11000 nM T27602 CX1WM9 21366579 IC50 > 11000 nM T27602 CA63IO 21706943 Ki = 320 nM T27602 C80JYP 21707001 Ki = 1200 nM T27602 C5JD2U 21707080 Ki = 200 nM T27602 CI0SJ2 21967345 Ki = 860 nM T27602 CK5I4A 21968289 Ki > 1600 nM T27602 CF4JN6 22010099 Ki = 132000 nM T27602 C7ZA4U 22010100 Ki = 138000 nM T27602 CFO41P 22010118 Ki = 20000 nM T27602 CA3I4Y 22280766 Ki > 5200 nM T27602 C4YL7S 22556963 Ki = 610 nM T27602 C9VXC8 22556983 Ki = 2400 nM T27602 C7SJ9B 22665658 IC50 = 27000 nM T27602 CMXF83 22665728 IC50 = 8000 nM T27602 CN3ZI2 22883539 Ki > 2900 nM T27602 CW8EH6 22883547 Ki > 2900 nM T27602 CA3N9L 22883564 Ki > 2900 nM T27602 C9DB7V 22883573 Ki > 2900 nM T27602 CVZ15N 22883583 Ki = 2900 nM T27602 C1R0UD 22883585 Ki = 2900 nM T27602 C13-JAN 22883594 Ki = 1800 nM T27602 C3VZ7S 23283289 Ki = 2000 nM T27602 CV5NL8 23283331 Ki = 1700 nM T27602 CSY57G 23646463 Ki = 420 nM T27602 C7E4SA 23646732 Ki = 700 nM T27602 C1Z9SX 24776379 Ki = 0.03 nM T27602 CQ6T4Z 43248030 Ki = 500034535 nM T27602 CTZ32N 43267452 Ki = 909913272.6 nM T27602 C2XLN7 44264885 Ki > 1600 nM T27602 CW4R8J 44264888 Ki > 4200 nM T27602 CT2V6S 44264889 Ki > 8000 nM T27602 CZDW40 44264920 Ki > 8000 nM T27602 C9RZ0O 44264921 Ki > 8000 nM T27602 CXQ1H9 44264935 Ki > 1600 nM T27602 C6O5VF 44264936 Ki > 1600 nM T27602 CVBG38 44264940 Ki > 8000 nM T27602 C63WPN 44264954 Ki > 4200 nM T27602 CB3AQ1 44264955 Ki > 4200 nM T27602 CGCI69 44264981 Ki > 8000 nM T27602 C78WPK 44264995 Ki > 4200 nM T27602 C01WIT 44265005 Ki > 8000 nM T27602 C1BP7E 44265006 Ki > 1600 nM T27602 CQNX29 44265034 Ki > 8000 nM T27602 C6OJ4I 44266844 Ki = 770 nM T27602 CB4ZN6 44266860 Ki = 420 nM T27602 C4LWN5 44266873 Ki = 580 nM T27602 CN5AV1 44266874 Ki = 0.27 nM T27602 CMCS75 44272530 Ki = 200 nM T27602 C6GRO0 44272532 Ki = 98 nM T27602 C65SNR 44272562 Ki = 69 nM T27602 C8CJI6 44272581 Ki = 500 nM T27602 CKZ6O0 44272690 Ki > 168 nM T27602 CT9XH1 44272744 Ki = 76.5 nM T27602 CB64EA 44272825 Ki = 16.6 nM T27602 CMD6Y8 44273648 Ki = 540000 nM T27602 CL7NY5 44274017 IC50 > 10000 nM T27602 CMG90C 44274089 IC50 > 10000 nM T27602 CO7Z3E 44274843 Ki = 3 nM T27602 CNZ83L 44274886 Ki = 5 nM T27602 C9UP2G 44274929 Ki = 120 nM T27602 C9WDV8 44274930 Ki = 6.9 nM T27602 C3U8OC 44274931 Ki = 32 nM T27602 C2U5SO 44274945 Ki = 410 nM T27602 C5VE6G 44275194 Ki = 3 nM T27602 CT2J0P 44275195 Ki = 10 nM T27602 C42RVS 44275227 Ki = 130 nM T27602 CQ12EP 44275238 Ki = 350 nM T27602 C3OM8S 44275239 Ki = 43 nM T27602 CGOH67 44275240 Ki = 73 nM T27602 CU52WR 44275243 Ki = 24 nM T27602 C2HO4D 44275249 Ki = 21 nM T27602 C1N5GM 44275254 Ki = 67 nM T27602 C9EKZ2 44275271 Ki = 320 nM T27602 C4TBU7 44275275 Ki = 15 nM T27602 C2D9YK 44275287 Ki = 73 nM T27602 CPBU68 44275289 Ki = 91 nM T27602 CL4D3K 44275297 Ki = 690 nM T27602 C3LS5P 44275326 Ki = 150 nM T27602 CHJC81 44275330 Ki = 190 nM T27602 C4SO5M 44275345 Ki = 430 nM T27602 CBA9T0 44275361 Ki = 140 nM T27602 CEWU09 44275365 Ki = 25 nM T27602 C7CK0J 44276899 IC50 = 1010 nM T27602 CVU1T9 44277085 IC50 = 156 nM T27602 C62TUQ 44277332 IC50 = 25 nM T27602 CHZ2Q4 44277564 IC50 = 6.4 nM T27602 C3H9CA 44281580 Ki = 630 nM T27602 CIUM69 44281581 Ki = 500 nM T27602 CAJB43 44281595 Ki = 340 nM T27602 C0T7OQ 44281652 Ki = 800 nM T27602 C9LK8J 44281725 Ki = 2800 nM T27602 C07TZM 44281805 Ki = 260 nM T27602 CSIQ87 44283615 IC50 = 1790 nM T27602 CHN6X0 44283616 IC50 = 1760 nM T27602 CML1T6 44283635 IC50 = 3 nM T27602 C2JMY1 44283808 Ki = 2100 nM T27602 CE0NG1 44283905 Ki = 3000 nM T27602 C7QU0Y 44283909 Ki = 350 nM T27602 CMFT95 44283921 Ki = 2200 nM T27602 CLGI45 44283936 Ki = 140 nM T27602 CAJX21 44283999 Ki = 890 nM T27602 C3WPL2 44284147 Ki = 940 nM T27602 C2NRA3 44284163 Ki = 1500 nM T27602 CMU9A4 44284541 IC50 = 188 nM T27602 CXK3M6 44284559 IC50 = 194 nM T27602 C36PXQ 44284752 IC50 = 2500 nM T27602 CQ82ZW 44286426 IC50 = 396 nM T27602 COPR02 44286428 IC50 = 160 nM T27602 CS5U7F 44286453 IC50 = 10.9 nM T27602 CPK5M6 44286709 Ki = 10000 nM T27602 CQ2A3R 44286878 Ki = 13000 nM T27602 CJP7K9 44286879 Ki = 45000 nM T27602 CRK53N 44286978 Ki = 26000 nM T27602 C7WU5K 44287028 Ki = 23000 nM T27602 CMA2Q6 44287039 Ki > 400000 nM T27602 C0DG5R 44287043 Ki = 260000 nM T27602 C0G3DY 44287647 Ki = 0.11 nM T27602 C9IC3S 44287667 Ki = 3.1 nM T27602 CQ75ND 44287668 Ki = 0.62 nM T27602 CDTY78 44287882 Ki = 0.7 nM T27602 C6QP1H 44287919 Ki = 70 nM T27602 C2N6JE 44287941 Ki = 7.4 nM T27602 CMY2L6 44287943 Ki = 13 nM T27602 CPD6J7 44287944 Ki = 25 nM T27602 CO95FJ 44287962 Ki = 35 nM T27602 CJH70N 44287992 Ki = 3.8 nM T27602 C7UQ9V 44287997 Ki = 0.64 nM T27602 CA02GU 44288104 Ki = 33 nM T27602 C4UQZ8 44288223 Ki = 4.7 nM T27602 C1NUA2 44288243 Ki = 5.3 nM T27602 CIG0D7 44288309 Ki = 4.2 nM T27602 CI0G4E 44289615 Ki = 20000 nM T27602 CZRH12 44290033 IC50 > 11000 nM T27602 CUY95P 44290108 IC50 > 11000 nM T27602 CS76AC 44290361 IC50 = 8300 nM T27602 CMY82L 44290376 IC50 > 20000 nM T27602 CHL9Y6 44290377 IC50 > 100000 nM T27602 CLDH85 44290378 IC50 = 620 nM T27602 CXO05N 44290379 IC50 > 200000 nM T27602 CNWI90 44290501 IC50 > 200000 nM T27602 CBE24K 44290502 IC50 = 9700 nM T27602 C94BSK 44290516 IC50 = 1700 nM T27602 CAXB95 44290518 IC50 > 50000 nM T27602 C49EPA 44290519 IC50 = 2200 nM T27602 C37IJH 44290520 IC50 = 2300 nM T27602 CU17NH 44290529 IC50 = 1700 nM T27602 CC8YQ3 44290530 IC50 = 66 nM T27602 CN04WY 44290542 IC50 = 36000 nM T27602 CF8JK0 44290543 Ki = 75 nM T27602 C05EYJ 44290555 IC50 = 30 nM T27602 C10ANS 44290556 IC50 = 8400 nM T27602 CO9JQ0 44290557 Ki > 2900 nM T27602 CY60EW 44290560 Ki = 130 nM T27602 C70XKC 44290569 Ki = 168 nM T27602 C9QS3I 44290584 Ki = 490 nM T27602 CUW14A 44290648 Ki = 36 nM T27602 C2UV6T 44290696 Ki = 300 nM T27602 C8LY1J 44290712 Ki = 230 nM T27602 C0SYK2 44290731 Ki = 38 nM T27602 CN6KP1 44290929 Ki > 2900 nM T27602 C0E1RV 44290930 Ki = 95 nM T27602 C8APX2 44290947 Ki = 90 nM T27602 CZ7PT1 44290965 Ki = 42 nM T27602 CTA7I1 44291034 Ki = 368 nM T27602 CH59WK 44291046 Ki = 51 nM T27602 CYFC04 44291049 Ki = 52 nM T27602 C7TNE0 44291050 Ki = 36 nM T27602 CC4RN5 44291077 Ki = 170 nM T27602 CA9TP1 44292003 Ki = 16000 nM T27602 C67GIO 44292022 Ki = 517000 nM T27602 C7DT0R 44292384 Ki > 10000 nM T27602 C2JQ3O 44292951 Ki = 1700 nM T27602 CW02PO 44292952 Ki = 2500 nM T27602 CL5VP0 44293219 Ki = 2600 nM T27602 C60GBH 44293221 Ki = 3400 nM T27602 CE0QR2 44293262 Ki = 1900 nM T27602 CC26FY 44293263 Ki = 20000 nM T27602 C0O2PG 44295723 Ki = 1300 nM T27602 C8AY9O 44296035 Ki = 42000 nM T27602 CQ51FN 44296074 Ki = 5000 nM T27602 C3DG0L 44296128 Ki = 440 nM T27602 CPF86Z 44296129 Ki = 3400 nM T27602 C38SDX 44296130 Ki = 8200 nM T27602 C1WU8B 44296135 Ki = 840 nM T27602 CZEX59 44311229 IC50 = 310 nM T27602 CKP5W7 44311564 IC50 = 62 nM T27602 C6TQ7D 44312627 IC50 = 5330 nM T27602 CTW03S 44312639 IC50 = 8780 nM T27602 C18PFJ 44312776 IC50 = 875 nM T27602 CGS74O 44312851 IC50 = 2570 nM T27602 CM5RQ6 44312966 IC50 = 6640 nM T27602 CGND24 44312967 IC50 = 521 nM T27602 CRN7I3 44313020 IC50 > 10000 nM T27602 C3X7VO 44313132 IC50 = 2900 nM T27602 C6G0NQ 44313284 IC50 = 2050 nM T27602 CYQ4I0 44313285 IC50 > 10000 nM T27602 C2D0JU 44313317 IC50 > 10000 nM T27602 CU8S5P 44313405 IC50 = 2400 nM T27602 CIQ1L7 44313498 IC50 = 4200 nM T27602 CF1S3C 44313499 IC50 = 6700 nM T27602 C0G3WT 44313500 IC50 = 8100 nM T27602 C8V3IH 44313932 IC50 > 2500 nM T27602 CT2ZD9 44314001 IC50 > 2500 nM T27602 CFXW28 44314002 IC50 = 2500 nM T27602 CM10DN 44314053 IC50 = 74.7 nM T27602 CCK1W8 44314117 IC50 > 2500 nM T27602 CT1X8J 44314118 IC50 = 163 nM T27602 C9LIC7 44314307 Ki = 0.28 nM T27602 C4JK6Z 44314435 Ki = 0.43 nM T27602 C9IN4E 44314967 IC50 = 470 nM T27602 C4Q9ZF 44315391 Ki = 95000 nM T27602 C87MBQ 44315392 Ki = 141000 nM T27602 C5CIL6 44315449 Ki = 17000 nM T27602 C2QOP6 44315450 Ki = 11000 nM T27602 C5WI0G 44315604 Ki > 1000000 nM T27602 CDW83E 44315605 Ki > 1000000 nM T27602 CIBE78 44315607 Ki = 237000 nM T27602 CZ3CY0 44315608 Ki = 162000 nM T27602 C07NBY 44315609 Ki > 1000000 nM T27602 C8DQ5R 44315610 Ki = 73000 nM T27602 C0Z7PI 44315635 Ki > 1000000 nM T27602 CJ5I9T 44315636 Ki > 1000000 nM T27602 C71UBD 44315637 Ki = 317000 nM T27602 C8UAJ1 44315641 Ki = 80000 nM T27602 CH7M1F 44315642 Ki = 121000 nM T27602 C0EG4V 44315643 Ki = 148000 nM T27602 C8MU4G 44315644 Ki > 1000000 nM T27602 C2U5HM 44315664 Ki = 15000 nM T27602 CPT78A 44315674 Ki = 262000 nM T27602 CEO18C 44315675 Ki = 131000 nM T27602 C25DGE 44315677 Ki = 17000 nM T27602 C45PHT 44315678 Ki = 4000 nM T27602 C5QUO9 44315743 Ki = 70000 nM T27602 CA8L4R 44315744 Ki = 182000 nM T27602 CPV7S5 44315758 Ki = 78000 nM T27602 CRVN48 44315788 Ki = 110000 nM T27602 C1QEV6 44315805 Ki = 126000 nM T27602 CB7Q2W 44315826 Ki = 20000 nM T27602 CPH5U7 44315831 Ki = 52000 nM T27602 CG3VB1 44315832 Ki = 54000 nM T27602 CZ8RS4 44315843 Ki = 72000 nM T27602 CUGF09 44315844 Ki = 56000 nM T27602 CX20QR 44315845 Ki = 44000 nM T27602 C4KF3H 44315846 Ki = 146000 nM T27602 CCXE57 44315848 Ki = 29000 nM T27602 C0IVD5 44315849 Ki = 274000 nM T27602 CU74AZ 44315850 Ki = 158000 nM T27602 C9QO7H 44315851 Ki = 165000 nM T27602 CF4I7B 44315852 Ki = 156000 nM T27602 CS6C5I 44315912 Ki = 156000 nM T27602 CF48NZ 44315913 Ki > 1000000 nM T27602 C6O5ZT 44315914 Ki > 1000000 nM T27602 C8VZ4J 44315915 Ki > 1000000 nM T27602 CZ6K5W 44316015 Ki = 111000 nM T27602 CUL40O 44316026 Ki = 171000 nM T27602 CAJ97K 44316048 Ki = 273000 nM T27602 CQ52SH 44316049 Ki = 38000 nM T27602 C1MRI0 44316050 Ki = 50000 nM T27602 CV38TK 44316051 Ki = 126000 nM T27602 CKWY45 44316065 Ki = 144000 nM T27602 C97NYB 44317783 IC50 = 1375 nM T27602 C5AK3D 44317785 IC50 = 52.2 nM T27602 CFCJ83 44318038 IC50 = 2500 nM T27602 CW2X9Z 44318052 IC50 = 2500 nM T27602 C90NPX 44318079 IC50 = 8700 nM T27602 CBQ0D2 44318098 IC50 = 18200 nM T27602 C57VSJ 44318156 IC50 = 14000 nM T27602 CK58VB 44318182 IC50 = 2 nM T27602 CV8IB4 44318218 IC50 = 90 nM T27602 C1C0UG 44318220 IC50 = 74800 nM T27602 CK5RC4 44318223 IC50 = 139 nM T27602 COV05F 44318305 IC50 = 26600 nM T27602 C7C8BZ 44319291 Ki > 2900 nM T27602 CEZ84L 44320397 IC50 = 40 nM T27602 CSK62O 44320493 IC50 = 135 nM T27602 CYT2Q4 44320495 IC50 = 110 nM T27602 CG36WH 44320752 IC50 = 27 nM T27602 CQ64CD 44320839 IC50 = 77 nM T27602 CK1EZ2 44320862 IC50 = 26 nM T27602 C7AMH4 44320876 IC50 = 75 nM T27602 CX73RG 44324726 Ki = 120 nM T27602 CMZ05T 44324727 Ki > 1200 nM T27602 CI5BY6 44324744 Ki > 1600 nM T27602 CWN4P7 44325526 Ki > 2900 nM T27602 C1MT8R 44325527 Ki > 2900 nM T27602 CBD24R 44325803 Ki = 55 nM T27602 CZW79L 44325865 Ki > 2900 nM T27602 C4Q8AC 44325938 Ki > 2900 nM T27602 C61VAC 44325939 Ki > 2900 nM T27602 CK92AD 44325940 Ki > 2900 nM T27602 C5TLH0 44325953 Ki > 2900 nM T27602 CHI47Q 44325959 Ki = 570 nM T27602 C1DES8 44325967 Ki > 2900 nM T27602 C5CLJ1 44325971 Ki = 230 nM T27602 CYOQ97 44325982 Ki > 2900 nM T27602 C3A2IO 44325983 Ki > 2900 nM T27602 CO2F4Z 44326181 Ki > 2900 nM T27602 CF92WZ 44326243 Ki = 140 nM T27602 C90VZO 44326339 Ki = 310 nM T27602 CAG6M5 44327046 Ki = 21500 nM T27602 CTDM97 44327484 Ki > 1200 nM T27602 C86YFO 44327490 Ki = 510 nM T27602 CE3UL6 44327872 Ki = 230 nM T27602 C5Q8SZ 44328328 IC50 = 2000 nM T27602 CWR3M9 44328445 IC50 = 18000 nM T27602 CY7G8N 44328503 IC50 = 205000 nM T27602 C51DLA 44328525 IC50 = 4000 nM T27602 CBO8W3 44328590 IC50 = 13000 nM T27602 CRPE62 44328622 IC50 = 6000 nM T27602 C26KJP 44330423 Ki = 8.4 nM T27602 C1Z5FA 44330631 Ki = 0.61 nM T27602 CK8FJ6 44330632 Ki = 21 nM T27602 CS1V3W 44330665 Ki = 2.8 nM T27602 CQX7A3 44330666 Ki = 18 nM T27602 CWV7X5 44330835 Ki = 1.1 nM T27602 C98KLH 44330847 Ki = 3.8 nM T27602 CSM3B6 44330879 IC50 = 1770 nM T27602 CVM21A 44330906 IC50 > 7930 nM T27602 CY72JW 44330907 IC50 > 10000 nM T27602 CA4Y1P 44330934 IC50 > 10000 nM T27602 C9KW3Q 44331002 IC50 > 10000 nM T27602 CJ9Y8Z 44331003 IC50 = 4810 nM T27602 CR7F8L 44331114 IC50 > 10000 nM T27602 C4NP5G 44331140 IC50 > 10000 nM T27602 CFK17Y 44331147 IC50 > 10000 nM T27602 C2BS5N 44331180 IC50 = 888 nM T27602 CF13OL 44331190 IC50 = 5640 nM T27602 CE69GW 44331194 IC50 = 2150 nM T27602 C3SU1R 44331210 IC50 > 10000 nM T27602 C0YOA6 44331389 IC50 = 0.5 nM T27602 CGL57V 44331419 IC50 = 220 nM T27602 C6OPK8 44331423 IC50 = 3300 nM T27602 CTB69R 44331436 IC50 = 33 nM T27602 C5M2LB 44333833 Ki = 180 nM T27602 C7Y8IG 44334488 Ki = 3 nM T27602 CHL01I 44334805 Ki = 12 nM T27602 C61CGV 44337884 IC50 = 9 nM T27602 C4EFA8 44337894 IC50 = 29 nM T27602 C0HP3T 44337899 IC50 = 64000 nM T27602 CH0K1J 44337917 IC50 = 19 nM T27602 CG6T9S 44337925 IC50 = 890 nM T27602 CA10BE 44337935 IC50 = 260 nM T27602 C4ATV2 44337945 IC50 = 14 nM T27602 C2AN5G 44337986 IC50 = 15 nM T27602 CTD5Q8 44338012 IC50 = 350 nM T27602 C5OVP7 44338032 IC50 = 180 nM T27602 C9P8UK 44338157 IC50 = 22200 nM T27602 C04MBF 44338376 IC50 = 250 nM T27602 CA1G6Q 44338381 IC50 = 5700 nM T27602 CI70HX 44338476 Ki = 7000 nM T27602 CKA1T3 44341287 IC50 = 1.36 nM T27602 CZ9BF5 44341288 IC50 = 11.6 nM T27602 C4XEK1 44341417 IC50 = 2.58 nM T27602 CNW1B2 44342560 IC50 = 11940 nM T27602 CM7G1U 44342634 IC50 = 7750 nM T27602 CQW48S 44342644 IC50 = 31600 nM T27602 CCYN38 44342736 IC50 = 8990 nM T27602 CC0Z8V 44343581 IC50 = 26.6 nM T27602 CW76HT 44343582 IC50 = 324 nM T27602 CD0TW8 44343615 IC50 = 166 nM T27602 C9NZE1 44343799 IC50 = 75 nM T27602 CAIZ35 44343800 IC50 = 20.38 nM T27602 C0W6EI 44343845 IC50 = 152 nM T27602 C46IGW 44343852 IC50 > 2500 nM T27602 C5H3NY 44343853 IC50 > 31.2 nM T27602 C40EHX 44343858 IC50 = 59.2 nM T27602 C91PVF 44343859 IC50 = 4.21 nM T27602 C4MS5Q 44343972 IC50 = 40.3 nM T27602 C3ZI7A 44343993 IC50 = 30 nM T27602 CMEI89 44343994 IC50 = 223 nM T27602 CEA17Z 44344039 IC50 = 74.5 nM T27602 CUO74X 44344054 IC50 = 160 nM T27602 CIG0Q2 44344067 Ki = 466000 nM T27602 CQ7R5F 44344069 Ki = 1300 nM T27602 CANQ97 44344083 Ki = 67000 nM T27602 C52JVD 44344096 Ki = 106000 nM T27602 CBTF46 44344097 Ki = 437000 nM T27602 C60GZW 44344100 IC50 = 111 nM T27602 CAJT87 44344125 Ki = 6200 nM T27602 C93EWF 44344138 Ki = 23000 nM T27602 C0B1CU 44344151 Ki = 6300 nM T27602 C6CDJ3 44344152 Ki = 14200 nM T27602 CREZ48 44344153 IC50 = 561 nM T27602 CRYS42 44344167 Ki > 1000000 nM T27602 CK9YA3 44344184 Ki = 1600 nM T27602 C1LS3Q 44344185 Ki = 252000 nM T27602 C3RBW8 44347347 Ki = 300 nM T27602 CAY34C 44347478 Ki = 2200 nM T27602 CT0QN1 44347480 Ki = 2200 nM T27602 CV6KA1 44347491 IC50 = 2500 nM T27602 C2EH3B 44347493 IC50 = 79.8 nM T27602 C65ORY 44347498 IC50 = 41.3 nM T27602 CN7L4W 44347532 IC50 = 135 nM T27602 C1UN9I 44347534 Ki = 890 nM T27602 CM3P8Z 44347559 IC50 = 247 nM T27602 CJ5A8E 44347561 IC50 = 143 nM T27602 C0V2FL 44347624 Ki = 1900 nM T27602 CTQ93K 44347853 Ki > 1600 nM T27602 CA7C9J 44347854 Ki > 1600 nM T27602 C7F6BG 44347997 Ki > 1600 nM T27602 C58MFB 44348077 IC50 > 10000 nM T27602 CJ1XO7 44348087 Ki > 1600 nM T27602 CQ8CK5 44348093 Ki = 69 nM T27602 C31JWA 44348108 Ki > 1600 nM T27602 C2M6TU 44348587 IC50 > 10000 nM T27602 CED0Q4 44348616 IC50 > 10000 nM T27602 CZI93S 44348618 IC50 > 10000 nM T27602 C94NSH 44348621 IC50 > 10000 nM T27602 CV5F9W 44348635 IC50 > 10000 nM T27602 C6QXM9 44348648 IC50 > 10000 nM T27602 CSY03Q 44350110 Ki = 38 nM T27602 CN5H9Q 44350175 Ki = 160 nM T27602 C87NXA 44350193 Ki = 16 nM T27602 C4Y3TQ 44350195 Ki = 81 nM T27602 C0Q7KU 44350214 Ki = 960 nM T27602 CK9BD0 44352629 Ki = 1900 nM T27602 C4Z7EM 44352695 Ki = 20900 nM T27602 CDLQ89 44354931 IC50 = 8800 nM T27602 CZG9E2 44354934 IC50 = 990 nM T27602 C7NWU8 44354935 IC50 = 18000 nM T27602 C5UJB8 44354936 IC50 = 2900 nM T27602 CRL78E 44354968 IC50 = 1800 nM T27602 CM73HF 44354971 IC50 = 2200 nM T27602 CVYF38 44354984 IC50 = 8200 nM T27602 CZDW93 44355000 IC50 = 1800 nM T27602 CG1VN6 44355001 IC50 = 18000 nM T27602 CL04TR 44355071 IC50 = 1600 nM T27602 C9U4BR 44355072 IC50 = 3900 nM T27602 CI4R1U 44355083 IC50 = 3300 nM T27602 CDON50 44355100 IC50 > 1000000 nM T27602 C8BC3Z 44358436 Ki > 2500 nM T27602 CPO39C 44358576 Ki = 140 nM T27602 C82XKL 44359703 IC50 = 16750 nM T27602 C29ANK 44359723 IC50 = 791 nM T27602 C4Y5HK 44359726 IC50 = 2500 nM T27602 CIKY14 44359730 IC50 = 74.5 nM T27602 C40POZ 44359735 IC50 = 1.36 nM T27602 C5P3UG 44359755 IC50 = 467 nM T27602 C5ES1X 44359805 IC50 = 147 nM T27602 C5CTA0 44359810 IC50 = 137 nM T27602 CSV16F 44359885 IC50 = 1.52 nM T27602 CD3R9Q 44359906 IC50 = 16.6 nM T27602 CERC69 44359907 IC50 > 2500 nM T27602 CMDB96 44360123 IC50 = 770 nM T27602 CN3TD7 44365378 IC50 = 16.4 nM T27602 CSN3E7 44365380 IC50 = 22.3 nM T27602 CY5ZU1 44365482 IC50 = 3.8 nM T27602 CW86PH 44365662 IC50 = 17.1 nM T27602 C4Y9ZT 44365668 Ki = 500034535 nM T27602 C1AI2B 44365669 Ki = 599791076.3 nM T27602 CZOU58 44365694 Ki = 699841996 nM T27602 CK87XR 44365721 Ki = 29991625.19 nM T27602 CR49PQ 44365722 Ki = 299916251.9 nM T27602 C5YT9W 44366105 Ki > 1600 nM T27602 CT1F2W 44366339 Ki > 2500 nM T27602 C39FZP 44372663 Ki = 1700 nM T27602 C9I0BE 44372667 Ki = 120 nM T27602 CQLA75 44372683 Ki = 3400 nM T27602 CKFN05 44372724 Ki = 2800 nM T27602 CTD36H 44372738 Ki = 4500 nM T27602 CI6MQ5 44372778 Ki = 650 nM T27602 CFH41R 44372839 Ki = 110 nM T27602 C9COY7 44372840 Ki > 1000000 nM T27602 C34AWY 44372863 Ki = 4300 nM T27602 CZE15A 44372864 Ki = 1800 nM T27602 C7X5BE 44372865 Ki = 3.2 nM T27602 C2E6TP 44372889 Ki = 900 nM T27602 C36XWM 44372903 Ki = 4.8 nM T27602 CJC73F 44374707 IC50 = 255000 nM T27602 C34XTM 44375987 IC50 = 0.8 nM T27602 CD0W7C 44376100 IC50 = 10.8 nM T27602 C0Y8QD 44376252 IC50 = 20.5 nM T27602 C5R2PM 44376328 IC50 = 20 nM T27602 CTZR83 44376339 Ki = 1100 nM T27602 CH95MO 44376405 Ki = 12600 nM T27602 C5VDG0 44376417 IC50 = 2 nM T27602 CG64YQ 44376426 IC50 = 33 nM T27602 CKI3R7 44376454 Ki = 3900 nM T27602 CSW71I 44376504 Ki = 3300 nM T27602 C7WTQ1 44376505 Ki = 3600 nM T27602 C51GQP 44376523 Ki = 5400 nM T27602 CA7GW4 44376525 Ki = 4100 nM T27602 CKHG50 44376548 Ki = 10000 nM T27602 CZ68PY 44376566 Ki = 6000 nM T27602 C41SQG 44376585 Ki = 7900 nM T27602 C1PK0O 44376651 Ki = 340 nM T27602 CXG42V 44376671 Ki = 16200 nM T27602 CXZP98 44376712 Ki = 460 nM T27602 CUFO93 44376713 Ki = 2200 nM T27602 CEKG07 44376754 Ki = 650 nM T27602 CQX98K 44376755 Ki = 5500 nM T27602 C2JKH1 44376756 Ki = 4900 nM T27602 CITM85 44376766 Ki = 17400 nM T27602 CV7I3K 44376788 Ki = 8500 nM T27602 CV5J1M 44376828 Ki = 12600 nM T27602 C6QG0C 44377053 Ki = 2100 nM T27602 C6A7VL 44377057 Ki = 2200 nM T27602 CI2GS0 44377287 IC50 = 147 nM T27602 C7W2GD 44377304 IC50 = 15 nM T27602 CP0V6X 44377320 IC50 = 145 nM T27602 C4KSG5 44377322 IC50 = 115 nM T27602 CH1NM4 44377327 IC50 = 412 nM T27602 CTP28F 44377331 IC50 = 25 nM T27602 C30VGP 44377425 IC50 = 75 nM T27602 CT0G2D 44377544 IC50 = 158 nM T27602 CK6I3F 44377546 IC50 = 537 nM T27602 CNUL43 44377548 IC50 = 211 nM T27602 CZBJ51 44377550 IC50 = 447 nM T27602 CHU5T4 44377558 IC50 = 33 nM T27602 CO7N6Y 44378546 Ki = 409000 nM T27602 C1WB3Q 44378759 Ki = 730300 nM T27602 CLXH02 44378887 Ki = 342000 nM T27602 CGL17Z 44379037 Ki > 100000 nM T27602 COH45E 44379112 Ki > 100000 nM T27602 CMW49N 44379117 Ki > 1000000 nM T27602 CWJ5E6 44379904 Ki = 3000 nM T27602 CJ0P4F 44379905 Ki = 2100 nM T27602 CY4HT3 44380201 Ki = 1500 nM T27602 CZ13VE 44380217 IC50 = 4300 nM T27602 CD36KV 44380417 Ki = 4 nM T27602 CI4RX8 44380662 IC50 = 24 nM T27602 CVG5S6 44380663 IC50 < 1 nM T27602 CC4MP1 44380667 Ki = 20 nM T27602 CC8DX1 44380674 IC50 = 160 nM T27602 CU98BT 44380699 IC50 = 12 nM T27602 CZ6NT9 44380722 IC50 = 2 nM T27602 C91WQC 44380740 IC50 = 8490 nM T27602 C2XH6Q 44381062 IC50 = 970 nM T27602 C3I2DC 44381063 IC50 = 18680 nM T27602 C8I5OP 44381104 IC50 = 14 nM T27602 CJ6M5B 44382389 IC50 = 257 nM T27602 CTF4N6 44382391 IC50 = 103 nM T27602 CAI65F 44382441 IC50 = 1220 nM T27602 C6LH5V 44383081 IC50 = 791 nM T27602 C9SD3E 44383242 Ki > 2900 nM T27602 C5PW9E 44383425 IC50 = 479 nM T27602 C43KTU 44383519 Ki > 2900 nM T27602 CNBG48 44383542 IC50 = 1220 nM T27602 C2IX5U 44383543 IC50 = 188 nM T27602 CBN31W 44384237 Ki > 15000 nM T27602 C5DAB6 44384238 Ki > 6000 nM T27602 CE5P9W 44384391 Ki = 140 nM T27602 C6IX3V 44384674 Ki = 300 nM T27602 CNB73E 44384879 Ki = 280 nM T27602 C6H0NF 44384928 Ki = 310 nM T27602 CJ01YE 44385090 Ki = 30 nM T27602 CV4N1P 44385091 Ki = 90 nM T27602 C1ZV8A 44385092 Ki = 20 nM T27602 C7U0HZ 44385205 Ki = 60 nM T27602 CTX13E 44385259 Ki = 670 nM T27602 CI91SG 44385260 Ki = 250 nM T27602 C4RV6U 44385263 Ki = 90 nM T27602 CHPL94 44385310 Ki = 690 nM T27602 C6VZ5Y 44385361 Ki = 1620 nM T27602 CPV5B7 44385418 Ki = 410 nM T27602 C8CE6A 44385432 Ki = 410 nM T27602 CG7LT1 44385488 IC50 > 11000 nM T27602 C94GZU 44385541 IC50 > 11000 nM T27602 C3T9XK 44385607 IC50 > 11000 nM T27602 CKY0P4 44385611 IC50 > 11000 nM T27602 CUS20V 44385673 IC50 > 11000 nM T27602 CZ8XL6 44385679 IC50 > 11000 nM T27602 CL5BA4 44385729 IC50 > 11000 nM T27602 C3DSN7 44385768 IC50 > 11000 nM T27602 C8USN9 44385769 IC50 > 11000 nM T27602 C2E8DS 44385771 IC50 > 11000 nM T27602 C2VFC6 44385772 IC50 > 11000 nM T27602 CN8V0W 44385779 IC50 > 11000 nM T27602 CBEA65 44385842 IC50 > 11000 nM T27602 C4XY8T 44385865 Ki = 510 nM T27602 CC9M7E 44385869 IC50 > 11000 nM T27602 C8WK4A 44385891 IC50 > 11000 nM T27602 C3D2CL 44385935 IC50 > 11000 nM T27602 CFPH43 44385967 Ki = 30 nM T27602 CW08OY 44385998 IC50 > 11000 nM T27602 CV6KG4 44386059 IC50 > 11000 nM T27602 CGU69V 44386179 IC50 > 11000 nM T27602 CS65LH 44386185 IC50 > 11000 nM T27602 CU0P5T 44386242 IC50 > 11000 nM T27602 CU9J0D 44386250 IC50 > 11000 nM T27602 C9G7QW 44386322 IC50 > 11000 nM T27602 C31CUG 44386326 IC50 > 11000 nM T27602 C2WCE4 44386371 IC50 > 11000 nM T27602 C52POK 44386417 IC50 > 11000 nM T27602 CRX1I9 44386418 IC50 > 11000 nM T27602 CIBD76 44386484 IC50 > 11000 nM T27602 C8ME4O 44386493 IC50 > 11000 nM T27602 CD4AH3 44386540 IC50 > 11000 nM T27602 CHAO48 44386542 IC50 > 11000 nM T27602 CLNO15 44386637 IC50 > 11000 nM T27602 C81IMH 44386642 IC50 > 11000 nM T27602 C8SYK9 44386783 Ki = 5000 nM T27602 C4JB0M 44386841 IC50 > 11000 nM T27602 C5MR1F 44386934 IC50 > 11000 nM T27602 CA45DZ 44387044 IC50 > 11000 nM T27602 C39LUW 44387104 IC50 > 11000 nM T27602 C2QD1K 44387206 IC50 > 11000 nM T27602 CN2GR5 44390800 Ki = 50 nM T27602 CW3G5V 44390801 Ki = 80 nM T27602 CTS5W9 44404049 IC50 > 400000 nM T27602 CC6A4Y 44453083 IC50 = 2.3 nM T27602 CW1GP4 44453663 IC50 = 3360 nM T27602 C8ZYV5 44453904 IC50 = 27400 nM T27602 CTF95R 44454022 IC50 = 24000 nM T27602 CS1TF7 44460215 IC50 = 969 nM T27602 CVU5G4 44460232 IC50 = 2500 nM T27602 CH61KG 44460246 IC50 = 538 nM T27602 C8SC7A 44460306 IC50 = 139 nM T27602 CXG8H0 44460987 Ki = 4800 nM T27602 CWND94 44461897 IC50 = 7000 nM T27602 CZ1YR4 44461912 Ki = 13.5 nM T27602 C13ZYL 44461991 IC50 = 29000 nM T27602 CX2LS5 44461992 IC50 = 9700 nM T27602 C38UKJ 44461994 IC50 = 18500 nM T27602 CF0N9S 44461996 IC50 = 42700 nM T27602 CPY92L 44462032 IC50 = 17000 nM T27602 C74KGD 44462047 IC50 = 91200 nM T27602 C8BH4N 44462081 IC50 = 2500 nM T27602 CL1TX8 44462086 IC50 = 9100 nM T27602 CXMW10 44462102 IC50 = 4800 nM T27602 C0K9TY 44462103 IC50 = 4100 nM T27602 CH3WY6 44462136 IC50 = 33400 nM T27602 CA8K6V 44462137 IC50 = 3800 nM T27602 C1B5XA 44462146 IC50 = 25000 nM T27602 C74CRB 44462147 IC50 = 3700 nM T27602 C2UR1M 44462161 IC50 = 4800 nM T27602 CQ31TR 44462179 IC50 = 8500 nM T27602 CU8Q5J 44462244 IC50 = 2300 nM T27602 C9Y8EN 44462296 IC50 = 21000 nM T27602 C1LG0F 44462297 IC50 = 45000 nM T27602 CWB04E 44462312 IC50 = 202 nM T27602 CS84NF 44462330 IC50 = 7800 nM T27602 CT6S5P 44462346 IC50 = 96 nM T27602 C5GR0E 44462347 IC50 = 15000 nM T27602 CDN1P2 44462348 IC50 = 7200 nM T27602 CVZW52 44537923 IC50 = 1600 nM T27602 CZ4JW1 45261445 Ki = 282 nM T27602 CN19RU 45261811 Ki = 100 nM T27602 CK7E3M 45264760 Ki = 1000 nM T27602 CJ5E2P 45265199 Ki = 6 nM T27602 C4YAJ7 46228924 IC50 > 10000 nM T27602 CY47OV 46878192 Ki > 1200 nM T27602 CQ2G6A 46878194 Ki = 214 nM T27602 C39CXL 46878195 Ki > 1200 nM T27602 CC6GE9 46878197 Ki = 40 nM T27602 CE79OB 46878198 Ki > 1200 nM T27602 CS07EW 46878199 Ki > 1200 nM T27602 C3HZP7 46878200 Ki = 27 nM T27602 CF5ZQ8 46878201 Ki > 1200 nM T27602 C7ICJ0 46878202 Ki > 1200 nM T27602 CQJR51 46878203 Ki = 0.045 nM T27602 C9BXU7 46878204 Ki > 1200 nM T27602 CXQL63 46878205 Ki > 1200 nM T27602 CR93NC 46878206 Ki > 1200 nM T27602 CX2L8G 46905375 Ki = 130 nM T27602 CTR32W 46905376 Ki = 57 nM T27602 CR6P1E 46905379 Ki = 190 nM T27602 CEDL20 49796469 Ki = 170 nM T27602 CS90ZF 49796473 Ki = 60 nM T27602 CHB03N 54252937 Ki > 2900 nM T27602 CE5A7B 60162406 Ki = 44 nM T27602 CA49UK 69520512 Ki > 5400 nM T27602 CJY20L 70686249 Ki = 198000 nM T27602 CNY4B7 70688369 Ki = 647000 nM T27602 C30ZKJ 71561420 Ki = 8.4 nM T27602 CD53RA 71716975 Ki > 120000 nM T27602 CSP5T2 71716976 Ki > 120000 nM T27602 C4FQ0W 73345765 Ki = 2.1 nM T27602 CCD54H 73345766 Ki = 23 nM T27602 CQF46R 73348759 Ki > 1200 nM T27602 CSQ41U 73348767 Ki = 1.4 nM T27602 CAJ7O5 73350148 Ki = 5000 nM T27602 C5VP6W 73350339 Ki = 2.3 nM T27602 CK45HD 73350340 Ki = 8.4 nM T27602 C60BNQ 73350342 Ki = 12 nM T27602 C4CD7U 73351857 Ki = 36 nM T27602 C60JSR 73353029 Ki = 1700000 nM T27602 C69BHN 73353326 Ki = 9.6 nM T27602 C26QPS 73353327 Ki = 4.2 nM T27602 C7DGZ9 73353328 Ki = 1.9 nM T27602 CA2P1B 73353330 Ki = 6.6 nM T27602 CD8M1N 73354683 IC50 = 5200 nM T27602 CNRW95 73354848 Ki = 35 nM T27602 COF2K0 73354849 Ki = 7.1 nM T27602 C3VFD6 73354850 Ki = 2.7 nM T27602 CL34CV 73354863 Ki = 5.6 nM T27602 C8N4RM 73356390 Ki = 4.8 nM T27602 CS7WY0 76313442 Ki = 150 nM T27602 CC2Q1D 76316954 Ki = 1400 nM T27602 C54OUH 76316955 Ki = 65000 nM T27602 C7QGZ9 76316957 Ki = 29 nM T27602 CQN23P 76324323 Ki = 8000 nM T27602 CP6HX3 76327889 Ki = 2400 nM T27602 C2MEC1 76327890 Ki = 35 nM T27602 CZDM90 76331536 IC50 = 550 nM T27602 CYD98M 76331537 Ki > 400 nM T27602 CL6X7D 76335180 IC50 = 0.6 ug.mL-1 T27602 C84POR 90664298 Ki = 5800 nM T27602 C7BX6R 90664760 Ki = 45 nM T27602 CBL46V 121488126 IC50 = 6 nM T27602 C3WC9Y 121488127 IC50 = 19 nM T27602 CE26HW 131955087 IC50 = 110 nM T27602 CD53CZ 135404951 Ki = 2200 nM T27602 C5XA6H 135407717 Ki = 18000 nM T27602 C0OX6T 135407736 Ki = 30000 nM T27602 C61XOA 135427245 Ki = 30000 nM T27602 C8WS4O 135443730 Ki = 9000 nM T27602 C3SMN4 135444666 IC50 = 283 nM T27602 CDT1C6 135452907 Ki = 6700 nM T27602 C3YT2M 135452929 Ki = 17000 nM T27602 CPN5I3 135452944 Ki = 40 nM T27602 C9KLD3 135455964 Ki > 2900 nM T27602 CJWC64 135462427 Ki = 305 nM T27602 C5O6JX 135469686 Ki = 80 nM T27602 C9XMA6 135469687 Ki = 110 nM T27602 CXS6B9 135471524 Ki = 6000 nM T27602 C2PFI8 135475618 Ki = 8500 nM T27602 CG2N5B 135484079 Ki = 90 nM T27602 CBE9G0 135490854 Ki = 18000 nM T27602 CPW07U 135493126 Ki = 580 nM T27602 CMQ6O0 135501618 Ki = 15000 nM T27602 CVA61N 135512760 Ki = 14000 nM T27602 CLFR21 135528485 Ki = 41000 nM T27602 CHEQ21 135528490 Ki = 4600 nM T27602 CL8PD0 135528527 Ki = 4000 nM T27602 CK97FT 135533257 Ki = 3300 nM T27602 CAD75F 135535997 Ki = 6500 nM T27602 C67TIA 135544099 IC50 = 2290 nM T27602 CCH49A 135544551 Ki = 3500 nM T27602 CKLD47 135544579 Ki = 16000 nM T27602 C8KNC4 135681488 Ki = 110 nM T27602 C6MZP7 135763271 Ki = 2200 nM T27602 C68GTN 135763273 Ki = 2300 nM T27602 C91UXW 135802775 Ki > 2900 nM T27602 CQD2Z1 135855944 Ki = 4.7 nM T27602 CMJ0B6 135962022 Ki ~ 2900 nM T27602 C9G7TE 135995982 Ki = 1300 nM T27602 CK36ZW 136029160 Ki = 240 nM T27602 CYQ70K 136053621 IC50 > 11000 nM T27602 C46VRO 136058172 Ki = 1400 nM T27602 C6Q4FB 136058174 Ki = 1400 nM T27602 C34UZI 136058175 Ki = 1600 nM T27602 CUX79V 136058176 Ki = 1900 nM T27602 CBY56D 136058177 Ki ~ 2900 nM T27602 C4YO6Q 136058178 Ki > 2900 nM T27602 CB39EK 136058180 Ki > 2900 nM T27602 C8PLB3 136058181 Ki > 2900 nM T27602 CSU6X4 136058182 Ki = 1400 nM T27602 C0Y3CA 136058183 Ki = 1500 nM T27602 C8IH1Z 136058184 Ki = 240 nM T27602 C4LG7S 136058185 Ki > 2900 nM T27602 CCX30L 136058186 Ki > 2900 nM T27602 C6KG8F 136058187 Ki = 1400 nM T27602 CHS25L 136058188 Ki = 1800 nM T27602 CSP4A7 136114639 Ki = 1200 nM T27602 CPK6X2 136198635 Ki = 1600 nM T27602 CRJ5S4 136198636 Ki > 2900 nM T27602 C7WE2G 136198637 Ki > 2900 nM T27602 C12UWY 136198638 Ki > 2900 nM T27602 CZM35V 145949585 Ki = 2.6 nM T27602 CKV37Z 145950098 Ki = 0.76 nM T27602 CI3XK5 145951517 Ki = 100 nM T27602 C4TRO0 145953377 Ki = 1.9 nM T27602 CC19VW 145957340 Ki = 0.87 nM T27602 C0A3MI 145959466 Ki = 49 nM T27602 CSBC71 146680900 IC50 = 11 nM T27602 C26NCB 155511048 IC50 = 3 nM T27602 CET60O 155514831 IC50 = 31000 nM T27602 CPUG37 155516479 Ki > 5400 nM T27602 CRW92X 155516645 IC50 = 5 nM T27602 C3W1DA 155526172 IC50 = 2100 nM T27602 C86HGK 155531857 IC50 = 110 nM T27602 CN07PE 155536057 IC50 = 100 nM T27602 CY3S0M 155537382 IC50 = 220 nM T27602 CCG68S 155539794 IC50 = 490 nM T27602 CAT09J 155541500 Ki > 5400 nM T27602 CURJ73 155545015 IC50 = 2 nM T27602 CW73AU 155546465 IC50 = 960 nM T27602 CWC8X9 155550748 IC50 = 8 nM T27602 CEX16I 155554542 IC50 = 160 nM T27602 CA37EY 155557358 IC50 = 330 nM T27602 CEI1Z4 155561184 IC50 = 110 nM T27602 C2GES3 2037 IC50 = 0.6 ug.mL-1 T27602 C2EIA8 44287957 Ki = 4.8 nM T27602 D02NHS 154118 Ki = 1800 nM T27602 D02XPB 23646462 Ki = 580 nM T27602 D03QAQ 9869498 Ki = 16 nM T27602 D03ZUM 6917805 IC50 = 14 nM T27602 D06MTX 1506 Ki = 23000 nM T27602 D07IBU 10696098 IC50 = 70 nM T27602 D07SGS 44292136 Ki = 568000 nM T27602 D08EUH 25113125 Ki > 1000000 nM T27602 D09OBJ 9872263 Ki = 3.1 nM T27602 D09YQM 9802488 IC50 = 4.5 nM T27602 D0A8WP 447732 Ki = 325 nM T27602 D0C1TS 44272875 Ki = 12.4 nM T27602 D0CT8A 23646461 Ki = 2000 nM T27602 D0F9YV 44365677 IC50 = 19.5 nM T27602 D0J2SM 296008 IC50 = 15300 nM T27602 D0K7YL 447476 Ki = 130 nM T27602 D0O0GT 44272797 Ki = 20.8 nM T27602 D0O1DU 25011732 Ki = 89000 nM T27602 D0S3VV 65526 Ki = 500034535 nM T27602 D0Y8QU 9869156 IC50 = 791 nM T16769 D0R1CR 6140 IC50 = 80200 nM T16769 D01NUR 118169620 IC50 = 2.8 nM T16769 D01YIF 135421197 IC50 > 10000 nM T16769 D03MXK 25022340 EC50 = 34 nM T16769 D07CLV 46940575 IC50 = 21 nM T16769 D09MIN 24737642 IC50 = 30 nM T16769 D0Q7AG 53240420 IC50 > 50000 nM T16769 D08UPQ 73603510 IC50 = 28 nM T16769 D08XOV 50913339 IC50 = 200 nM T16769 D0Q1XF 72710867 IC50 = 4 nM T16769 D0YN1X 71661892 Ki < 1 nM T16769 D05HSW 3218 Ki = 400 nM T16769 C0NJ2B 645025 IC50 = 1540 nM T16769 CRM9S6 674647 IC50 = 9810 nM T16769 CN06WE 685663 IC50 = 12800 nM T16769 C6ITY8 821411 Ki = 10400 nM T16769 C5UAR2 910374 IC50 = 6690 nM T16769 C83UKT 1223927 IC50 = 3990 nM T16769 CAX45S 3332652 IC50 = 8070 nM T16769 CW7YG3 3724041 IC50 = 810 nM T16769 C5ND2X 4369343 EC50 = 290 nM T16769 CC49SG 5316673 IC50 > 100000 nM T16769 CVJ68Z 5496538 IC50 = 400 nM T16769 CCD3J2 6918762 EC50 = 310 nM T16769 CE1Q0I 7019981 IC50 = 1200000 nM T16769 C0SWR7 10181236 IC50 = 56 nM T16769 C2IAF0 10222526 IC50 = 0.017 nM T16769 C83DPY 11151918 Ki = 4410 nM T16769 CG51SF 11176463 Ki = 1270 nM T16769 C4FEH8 11176734 Ki = 150 nM T16769 C17WQK 11178892 Ki = 1300 nM T16769 CMR39J 11190107 Ki = 60 nM T16769 CHGD18 11200722 Ki = 290 nM T16769 CW8CH5 11225031 Ki = 25 nM T16769 C4TZX5 11258581 Ki = 180 nM T16769 CFH7I5 11280887 Ki > 100000 nM T16769 C3KXC6 11317764 Ki = 28 nM T16769 C3UR2G 11351754 Ki = 24 nM T16769 CUG45Z 11395933 EC50 = 1260 nM T16769 C7N1KQ 11417324 Ki = 2450 nM T16769 CL2SN7 11417422 Ki = 150 nM T16769 C4H7EU 11450670 Ki = 13400 nM T16769 C0KD5Z 11475093 Ki = 220 nM T16769 CFXK28 11497354 Ki = 140000 nM T16769 CWZ8F7 11503417 IC50 = 1000 nM T16769 CM2IF7 11518553 Ki = 61 nM T16769 COHA56 11523380 Ki = 180 nM T16769 C67NHR 11562245 Ki = 14400 nM T16769 C2W7FX 11564993 Ki = 710 nM T16769 CA2Z5Y 11705765 Ki = 160 nM T16769 C87DVG 11765457 IC50 > 10400 nM T16769 C9KGH4 13224102 IC50 = 390 nM T16769 C2DLT9 16099367 Ki = 29000 nM T16769 CY3RV2 17756618 IC50 <= 1 nM T16769 CG19LI 23342610 IC50 = 14100 nM T16769 C4BS1H 23646334 Ki = 4900 nM T16769 CU35OX 23646335 Ki = 1200 nM T16769 C3EBC4 23646336 Ki = 68000 nM T16769 C3HQ6X 23646337 Ki = 81 nM T16769 CV8JE5 23646338 Ki = 4150 nM T16769 CY6FW5 23646339 Ki = 54000 nM T16769 CGV7U5 23646340 Ki = 1250 nM T16769 CUB57D 23646341 Ki = 1300 nM T16769 C7VR6X 23646342 Ki = 480 nM T16769 CMHO78 23646343 Ki = 380 nM T16769 CBM94F 23646361 Ki = 580 nM T16769 C5RV8Q 24754887 IC50 = 376 nM T16769 C8XJG1 24754961 Ki > 10000 nM T16769 C9N5YA 25011737 IC50 = 270 nM T16769 CF52WX 25011738 IC50 = 110 nM T16769 CO8K9S 25058143 IC50 = 86 nM T16769 C7XTN2 25138055 Ki = 30 nM T16769 CJ2VZ4 25138056 Ki = 18 nM T16769 C29PBM 25138057 Ki = 1200 nM T16769 CLO6Y8 25138058 Ki = 690 nM T16769 CSW2C4 25138059 Ki = 100 nM T16769 CB7V2M 25138060 Ki = 29000 nM T16769 C3P5EA 25138061 Ki = 14 nM T16769 C1ZEC7 25138062 Ki = 39 nM T16769 CLUP32 25138063 Ki = 759 nM T16769 CGS90Z 25138064 Ki = 47 nM T16769 C9U0DW 25138065 Ki = 67 nM T16769 C0J8QZ 25138066 Ki = 856 nM T16769 CEQ23J 25138067 Ki = 32870 nM T16769 C0JM7N 25138068 Ki = 12970 nM T16769 CPN8E5 25138069 Ki = 14 nM T16769 CWH17B 25138070 Ki = 209 nM T16769 C5MZ8T 25138071 Ki = 15 nM T16769 C0BJQ6 25173661 Ki = 67300 nM T16769 CSD59K 25173742 EC50 = 9280 nM T16769 CW4U0R 25180313 Ki = 51 nM T16769 C2SWF7 25195345 Ki = 570 nM T16769 C46SKW 25195346 Ki = 140 nM T16769 C2SL1P 25199552 Ki = 5620 nM T16769 CJ6E3C 25199554 Ki = 440 nM T16769 C61JBK 25199558 Ki = 590 nM T16769 CAL8M3 25209021 Ki = 3.9 nM T16769 CD29TU 25209022 Ki = 31 nM T16769 CGB36H 25218664 Ki = 210 nM T16769 C0DG7M 25218665 Ki = 190 nM T16769 CZ7T1V 25218666 Ki = 110 nM T16769 C29LKB 25218667 Ki = 1200 nM T16769 C81KNV 25218668 Ki = 500 nM T16769 C8HTW7 25218669 Ki = 8100 nM T16769 C8A0SB 25218670 Ki = 1800 nM T16769 CE41BP 25218671 Ki = 490 nM T16769 CEH14K 25218672 Ki = 1200 nM T16769 CHRE60 25218673 Ki = 1800 nM T16769 C6QL1R 25218674 Ki = 14300 nM T16769 C6RX3C 25218675 Ki = 1500 nM T16769 C1D5UY 25218676 Ki = 8600 nM T16769 CY4X3Z 25218677 Ki = 640 nM T16769 CR2LH1 25218678 Ki = 330 nM T16769 CP97QZ 25218679 Ki = 580 nM T16769 C7O0GJ 25218680 Ki = 5900 nM T16769 CH2F6N 25218681 Ki = 1500 nM T16769 CQPR85 25218682 Ki = 3000 nM T16769 CO10GL 25218683 Ki = 1600 nM T16769 C98BAU 25241634 Ki = 20070 nM T16769 C0W4PR 25241638 Ki = 120 nM T16769 CB5JZ4 25241640 Ki = 55 nM T16769 CS2G4D 25241656 Ki = 800 nM T16769 CHU2G3 25241658 Ki = 700 nM T16769 CXM52Z 25241666 Ki = 1910 nM T16769 C1IN4U 25241674 Ki = 390 nM T16769 CC6M7P 25241676 Ki > 39000 nM T16769 C40ZJB 25241680 Ki = 6070 nM T16769 C3L2AZ 25241682 Ki = 1400 nM T16769 CZ6JI9 25241691 Ki > 39000 nM T16769 CG10SZ 44176335 Ki = 2290 nM T16769 CIH9R3 44176337 Ki = 740 nM T16769 CL7EV1 44176339 Ki = 3040 nM T16769 CA8SJ6 44176341 Ki = 1740 nM T16769 CHC45V 44176343 Ki = 4540 nM T16769 C98KCZ 44176345 Ki = 2380 nM T16769 CTL67E 44176347 Ki = 640 nM T16769 CKZN29 44178407 IC50 = 14400 nM T16769 CP2Y6L 44182153 Ki = 350 nM T16769 CN3RB2 44182164 Ki = 650 nM T16769 C9NET8 44182176 Ki = 3650 nM T16769 CI8A1M 44182204 Ki = 3000 nM T16769 CI74QR 44182206 Ki = 1830 nM T16769 CY89SV 44182234 Ki = 660 nM T16769 CXAJ15 44182248 Ki = 1700 nM T16769 CTZ43W 44182250 Ki = 13140 nM T16769 C65XAD 44182256 Ki = 5460 nM T16769 CLWX45 44182258 Ki = 420 nM T16769 CD6I2H 44182260 Ki = 1290 nM T16769 C51PDE 44182262 Ki = 7200 nM T16769 C23JAM 44182264 Ki = 2550 nM T16769 CAJ47B 44182266 Ki = 1400 nM T16769 C35PGO 44182270 Ki = 4750 nM T16769 C48DHY 44182272 Ki = 8180 nM T16769 CA9D1W 44182274 Ki = 540 nM T16769 C5XC7D 44182276 Ki = 4940 nM T16769 CW6S2R 44229023 Ki = 1940 nM T16769 C1TA3I 44229037 Ki = 1880 nM T16769 CYO7P6 44229049 Ki = 3780 nM T16769 CY6IW9 44237042 IC50 = 200 nM T16769 C7N2HD 44237043 IC50 = 100 nM T16769 CSD8H1 44237044 IC50 = 450 nM T16769 CRPI49 44237045 IC50 = 320 nM T16769 CP1O5M 44237047 IC50 = 220 nM T16769 C0MF5P 44237048 IC50 = 4400 nM T16769 C1M7UE 44237049 IC50 = 240 nM T16769 C1QIE9 44237050 IC50 = 72 nM T16769 CY8FG6 44237051 IC50 = 650 nM T16769 C2E8OW 44237052 IC50 = 110 nM T16769 C6JDH9 44237053 IC50 = 110 nM T16769 CI2VK3 44237054 IC50 = 430 nM T16769 CR13NF 44237055 IC50 = 190 nM T16769 CS7I1D 44237056 IC50 = 110 nM T16769 CTEK15 44237057 IC50 = 240 nM T16769 C7Q4MH 44237058 IC50 = 510 nM T16769 CHR6Q2 44237059 IC50 = 190 nM T16769 C6CAK9 44237060 IC50 = 97 nM T16769 CMIH96 44237061 IC50 = 330 nM T16769 CJI4S9 44237062 IC50 = 54 nM T16769 CT9V5Y 44237063 IC50 = 240 nM T16769 CPG01O 44237064 IC50 = 54 nM T16769 CJ14RG 44237065 IC50 = 240 nM T16769 C5A7LH 44237066 IC50 = 85 nM T16769 C21XJR 44237067 IC50 = 70 nM T16769 CM6P2O 44237068 IC50 = 100 nM T16769 CJBR30 44396367 EC50 > 100000 nM T16769 CZ5I6X 44419748 Ki = 580 nM T16769 C38XKG 44460458 IC50 = 2800 nM T16769 C73UTK 44460459 IC50 = 570 nM T16769 C0AOS8 44589550 Ki = 14 nM T16769 C03TDR 44589551 Ki = 274 nM T16769 CCJT16 44590154 Ki = 4470 nM T16769 C3JR8F 44590155 Ki = 1410 nM T16769 CN0S1G 44590212 Ki > 100000 nM T16769 CAMK67 44590213 Ki = 43110 nM T16769 C7VT1X 44590214 Ki = 2330 nM T16769 CHVU50 44590215 Ki = 350 nM T16769 CO8G3P 44596256 IC50 = 27 nM T16769 CQY48M 44820626 Ki = 68000 nM T16769 C0E9LP 44820627 Ki = 36000 nM T16769 CA0UN2 45102735 Ki = 5580 nM T16769 CGKZ14 45263178 Ki = 350 nM T16769 CS40DG 45263184 Ki = 22400 nM T16769 CR0QT8 45263189 Ki = 4470 nM T16769 CYE95J 45263207 Ki > 100000 nM T16769 C5Q2IJ 45263221 Ki = 290 nM T16769 CY8O4N 45263222 Ki > 100000 nM T16769 C0TOA3 45263227 Ki = 1410 nM T16769 CE3L0W 45263230 Ki = 43110 nM T16769 CTH45I 45265670 Ki = 2330 nM T16769 C6H9LW 45265687 Ki > 100000 nM T16769 CK1RP4 45482532 IC50 = 600 nM T16769 CYG52W 45482547 IC50 = 120 nM T16769 CO83VD 45482548 IC50 = 55 nM T16769 CE83CZ 45482552 IC50 = 70 nM T16769 CO4W6H 45482560 IC50 = 75 nM T16769 CC9X5K 45482572 IC50 = 110 nM T16769 CDYU05 45482573 IC50 = 100 nM T16769 C69NUX 45482574 IC50 = 35 nM T16769 CSHM86 45487863 Ki = 37000 nM T16769 C3XU7D 46830176 Ki = 260000 nM T16769 C96OTK 46830178 IC50 = 0.43 nM T16769 CECL56 46830179 IC50 = 1.3 nM T16769 CL75NA 46883825 Ki = 31000 nM T16769 C2QPO5 46883826 Ki = 38000 nM T16769 CXT0Z7 46883827 Ki = 31000 nM T16769 CL3QR5 46883828 Ki = 31000 nM T16769 C6HNB8 46883881 Ki = 940000 nM T16769 CF2O4P 46883882 Ki = 190000 nM T16769 C6O1UC 46883883 Ki = 150000 nM T16769 C7JAQ0 46883921 Ki = 50000 nM T16769 CKUQ91 46883922 Ki = 60000 nM T16769 CW1PR3 46883923 Ki = 160000 nM T16769 C3SZP1 46883924 Ki = 55000 nM T16769 C8Z2MB 46883992 Ki = 58000 nM T16769 C8RBO6 46883993 Ki = 46000 nM T16769 CH92NU 46883994 Ki = 49000 nM T16769 CN0P3Q 46884021 Ki = 45000 nM T16769 C1DS6K 46884022 Ki = 41000 nM T16769 C90AVJ 46884023 Ki = 73000 nM T16769 C49JKQ 46884084 Ki = 51000 nM T16769 CPB9H7 46884085 Ki = 37000 nM T16769 CD7AG0 46884409 Ki = 190000 nM T16769 CF3QO9 46884410 Ki = 68000 nM T16769 CLZ07E 46884435 Ki = 35000 nM T16769 C2GB8Y 46884436 Ki = 19000 nM T16769 C40MQS 46884474 Ki = 75000 nM T16769 C8Q0RI 46884475 Ki = 130000 nM T16769 CE62KI 46884476 Ki = 100000 nM T16769 C0E5CW 46884477 Ki = 120000 nM T16769 C8RL0W 46884520 Ki = 47000 nM T16769 CM1D9E 46884521 Ki = 24000 nM T16769 C9X6JF 46884522 Ki = 35000 nM T16769 C59USH 46884523 Ki = 32000 nM T16769 C8RDC3 46888403 IC50 = 481 nM T16769 CP40QG 46929436 Ki = 108 nM T16769 CQ0A5I 46929438 Ki = 305.2 nM T16769 C5FK8W 46929440 Ki = 36 nM T16769 C1TIK8 46930628 Ki = 320.3 nM T16769 CVC3T5 46930723 Ki = 330.6 nM T16769 CQ3YK4 49789910 Ki = 2430 nM T16769 CN7I1W 49866703 Ki = 67 nM T16769 CD1G0B 50913340 IC50 = 240 nM T16769 CNQO70 52951104 Ki = 25.9 nM T16769 C30GIF 53237922 Ki = 5 nM T16769 CW7AF2 53238154 Ki = 3 nM T16769 C5JPH2 53238155 Ki = 1.5 nM T16769 CW71DY 53238387 Ki = 2 nM T16769 C16JNG 53238388 Ki = 4 nM T16769 C3IPJ4 53238615 Ki = 2 nM T16769 CH0L8C 53238616 Ki = 2 nM T16769 CF83PC 53238842 Ki = 1 nM T16769 C2HB0C 53238843 Ki = 1 nM T16769 C7SR2W 53239063 Ki = 1 nM T16769 CM46PV 53239064 Ki = 3 nM T16769 CNFD80 53239285 Ki = 4 nM T16769 CCL6I5 53239286 Ki = 88 nM T16769 C79PKU 53318805 Ki = 270 nM T16769 C3F7PD 53325387 IC50 = 280 nM T16769 CBIM49 56590676 IC50 = 1520 nM T16769 CK1NJ3 56590677 IC50 = 560 nM T16769 CO2HN7 56662840 Ki = 440 nM T16769 CIH4K7 56666366 Ki = 29880 nM T16769 CS65QR 56669774 Ki = 660 nM T16769 CT87XB 56679934 Ki = 1050 nM T16769 C61NHL 56945169 Ki = 2 nM T16769 C2WXP5 56945170 Ki = 2 nM T16769 C7YW1J 56945269 Ki = 3 nM T16769 CR7TD9 56945270 Ki = 2 nM T16769 CAD3P5 56945392 Ki = 1 nM T16769 CDYL09 56945393 Ki = 5 nM T16769 C7X1ZF 56946798 Ki = 3 nM T16769 C05JAE 56946799 Ki = 2 nM T16769 C8IWF7 57345674 IC50 = 111 nM T16769 CO9N3Z 57391385 IC50 = 47 nM T16769 CIP23W 57391386 IC50 = 41 nM T16769 C9FIB5 57391387 IC50 = 198 nM T16769 C6QHW5 57393149 IC50 = 47 nM T16769 CN0AF2 57396041 IC50 = 365 nM T16769 CXS64P 57396647 IC50 = 57 nM T16769 CI9MC4 57397789 IC50 = 650 nM T16769 C9G7YF 57398349 IC50 = 52 nM T16769 C8WZ1A 57400074 IC50 = 58 nM T16769 CHD41O 57400075 IC50 = 57 nM T16769 CG4B9T 57400076 IC50 = 53 nM T16769 C5N4FG 57400077 IC50 = 44 nM T16769 C9Q5WO 57400078 IC50 = 65 nM T16769 C6ZY0D 57400338 IC50 > 8000 nM T16769 C9IB0C 57401812 IC50 = 58 nM T16769 CZP8Q6 57401885 IC50 = 52 nM T16769 C9CRY4 57401886 IC50 = 78 nM T16769 CKU4F8 57403521 IC50 = 57 nM T16769 CESB84 57403599 IC50 = 181 nM T16769 COY56U 57522797 Ki = 35 nM T16769 C5F1MI 57522798 Ki = 430 nM T16769 CFE7J6 57522799 Ki = 190 nM T16769 CXQ63N 57522923 Ki = 7600 nM T16769 C8RN2I 57522924 Ki = 800 nM T16769 C2PFD7 57522925 Ki = 410 nM T16769 CH2IN5 57522926 Ki = 700 nM T16769 CE6SU4 57689264 Ki = 2 nM T16769 C62ZCQ 57689338 Ki = 1.5 nM T16769 CF89OA 58137904 IC50 = 120 nM T16769 C3KDR0 58609608 IC50 = 108.2 nM T16769 C1C7ML 59542215 IC50 = 5.3 nM T16769 CJL17T 60198193 IC50 = 18 nM T16769 C3QS0C 60198300 IC50 = 23 nM T16769 C16DYA 60198985 IC50 = 19 nM T16769 CW9U7M 66972432 IC50 = 120 nM T16769 CTYP01 66972671 IC50 = 190 nM T16769 CZI6S5 66972777 IC50 = 520 nM T16769 C06KWB 66972973 IC50 = 350 nM T16769 CK0FP7 66972990 IC50 = 300 nM T16769 CQ9Y8K 66972994 IC50 = 480 nM T16769 CTKN28 66973039 IC50 = 140 nM T16769 C0VG8C 66973046 IC50 = 650 nM T16769 CR9CO4 66973072 IC50 = 470 nM T16769 CKQ68O 66973165 IC50 = 410 nM T16769 CAD24O 66973224 IC50 = 1300 nM T16769 C0R9TP 66973397 IC50 = 1400 nM T16769 CQ1O6Z 66973400 IC50 = 240 nM T16769 COQ52M 70678411 IC50 <= 1 nM T16769 CM65DI 70980530 EC50 = 5.1 nM T16769 CO8YK2 70981017 EC50 = 140 nM T16769 C63JLP 71450435 IC50 = 3.9 nM T16769 C9BCY8 71452258 IC50 <= 1 nM T16769 CL31QP 71452260 IC50 <= 1 nM T16769 C9QF2G 71452262 IC50 = 5.9 nM T16769 CCGT91 71452264 IC50 = 15.5 nM T16769 CS4V9B 71452266 IC50 = 3.2 nM T16769 CM14JU 71454062 IC50 <= 1 nM T16769 CL3KX5 71454063 IC50 = 3.3 nM T16769 CQ8R3E 71454065 IC50 = 157 nM T16769 CZR6J5 71454067 IC50 = 1.6 nM T16769 C4JXM9 71454115 IC50 = 4.4 nM T16769 C90KFN 71457579 IC50 = 15.5 nM T16769 CG8X3Z 71457581 IC50 = 8.4 nM T16769 C82EPD 71457647 IC50 <= 1 nM T16769 C24OXD 71459481 IC50 <= 1 nM T16769 CTV86H 71459483 IC50 = 16.2 nM T16769 CMKI17 71459485 IC50 <= 1 nM T16769 CCS3R8 71461288 IC50 <= 1 nM T16769 CSGH36 71463006 IC50 <= 1 nM T16769 CQO9H5 71471883 IC50 = 9800 nM T16769 C9XW7O 71471946 IC50 = 46000 nM T16769 C6VW0X 71471950 IC50 = 51000 nM T16769 C3A9UH 71471953 IC50 = 59000 nM T16769 C5HTZ1 71472009 IC50 = 5500 nM T16769 CP13OU 71472011 IC50 = 5900 nM T16769 C14SJI 71472075 IC50 = 4100 nM T16769 CEH3B5 71472080 IC50 = 7700 nM T16769 C7QZX1 71472243 IC50 = 1500 nM T16769 CZ8DF4 71661893 Ki = 1.7 nM T16769 CB0O2T 71662077 Ki < 1 nM T16769 COCI81 71662078 Ki = 0.7 nM T16769 CNU16X 71662256 Ki < 1 nM T16769 CJRL34 71662257 Ki = 1.7 nM T16769 C2UM5A 71662420 Ki = 4.5 nM T16769 CVZK59 71662421 Ki < 1 nM T16769 CW4G0O 71662584 Ki < 1 nM T16769 C8AY6G 71662585 Ki = 1.3 nM T16769 C8P7YS 71713794 Ki = 780 nM T16769 C93WIS 71713796 Ki = 2020 nM T16769 CQ38NU 71713797 Ki = 670 nM T16769 C8O5YQ 71713798 Ki = 1130 nM T16769 CY2F6V 71713955 Ki = 2050 nM T16769 CJD9M4 71713956 Ki = 530 nM T16769 CTJ7H1 71714106 Ki = 4670 nM T16769 C2K0CS 71819719 IC50 = 6 nM T16769 C26SGQ 71819720 IC50 = 18 nM T16769 CV5FZ2 72711021 IC50 = 2770 nM T16769 CB41XI 72711023 IC50 = 6750 nM T16769 CK4T9G 72711025 IC50 = 2230 nM T16769 C8AJW5 72711027 IC50 = 150 nM T16769 CE5TM6 72711029 IC50 = 58 nM T16769 CZ0RU4 72711249 IC50 = 24800 nM T16769 C3SGZ4 72711251 IC50 = 8 nM T16769 CA6U8Q 72711253 IC50 = 27000 nM T16769 C7I9ZM 72711255 IC50 = 24300 nM T16769 CJF4B2 72711479 IC50 = 6 nM T16769 CNA70E 72711481 IC50 = 25700 nM T16769 CB09LR 72711483 IC50 = 22 nM T16769 CO5E7S 72711485 IC50 = 35 nM T16769 C2LCM8 72711720 IC50 = 5 nM T16769 C95UWO 72711722 IC50 = 7 nM T16769 C4O2MG 72711724 IC50 = 45900 nM T16769 C7PH3X 72711926 IC50 = 6 nM T16769 C6NOU0 72711928 IC50 = 6 nM T16769 CY4F2O 72711930 IC50 = 15 nM T16769 CJM96S 72711932 IC50 = 9 nM T16769 CQ72YG 72712127 IC50 = 10 nM T16769 C3UF4Z 72712129 IC50 = 9 nM T16769 C8WCQ4 72712131 IC50 = 19 nM T16769 C97PKX 72712133 IC50 = 58 nM T16769 CRO41V 72712330 IC50 = 5490 nM T16769 C95IJY 72712332 IC50 = 13800 nM T16769 CTI89S 72712334 IC50 = 4310 nM T16769 CD8GI6 72712336 IC50 = 1470 nM T16769 CK8BE1 72712338 IC50 = 702 nM T16769 CO4W7L 72712340 IC50 = 486 nM T16769 CXLI39 72712342 IC50 = 182 nM T16769 CP5NK4 72712344 IC50 = 83 nM T16769 C06CSU 72712346 IC50 = 32 nM T16769 CEPF37 72712559 IC50 = 249 nM T16769 C86TYE 72712561 IC50 = 194 nM T16769 CPG40K 72712563 IC50 = 1910 nM T16769 C7YKB8 72712565 IC50 = 31600 nM T16769 C2LUR6 72712567 IC50 = 104 nM T16769 CBL6M3 72712570 IC50 = 10 nM T16769 CTQ42C 72712572 IC50 = 51 nM T16769 CRL92T 72712769 IC50 = 81 nM T16769 CX8K7H 72712771 IC50 = 101 nM T16769 CB68YH 72712969 IC50 = 65 nM T16769 CS9D3G 72712971 IC50 = 48500 nM T16769 C8TD7A 72712973 IC50 = 36200 nM T16769 CF7BR8 72713167 IC50 = 22800 nM T16769 C6D3GW 72713169 IC50 = 569 nM T16769 CVA91J 72713170 IC50 = 183 nM T16769 CE37QK 72713171 IC50 = 32 nM T16769 C2C6XL 72713606 IC50 = 4390 nM T16769 CHD69M 72713610 IC50 = 383 nM T16769 C7A5EW 72714054 IC50 = 22 nM T16769 C7SZ3V 72714058 IC50 = 45 nM T16769 CY02QS 72714288 IC50 = 928 nM T16769 C24PBI 72714290 IC50 = 611 nM T16769 C81VNI 72714293 IC50 = 4360 nM T16769 CM85PO 72714295 IC50 = 2620 nM T16769 C5RD2F 72736709 IC50 = 62 nM T16769 CEK93U 72736862 IC50 = 220 nM T16769 C47KWN 72736863 IC50 = 140 nM T16769 CNAY12 73506219 IC50 = 17 nM T16769 C8QPX7 73507318 IC50 = 10 nM T16769 CKS45Y 73508005 IC50 = 2.9 nM T16769 C4K3BG 73508016 IC50 = 4.3 nM T16769 CETB68 73603641 IC50 = 10 nM T16769 C1A9ME 73672184 IC50 = 5.8 nM T16769 CJ38WP 73672428 IC50 = 3.5 nM T16769 CVOY02 73672545 IC50 = 16 nM T16769 CN3A1V 73672620 IC50 = 7.4 nM T16769 CALJ56 73672900 IC50 = 18 nM T16769 C8T2AC 73672902 IC50 = 12 nM T16769 C76XRT 73673026 IC50 = 30 nM T16769 CX95NQ 73673152 IC50 = 14 nM T16769 CPVS10 73673158 IC50 = 7.5 nM T16769 CF9GW8 73673640 IC50 = 47 nM T16769 C87QOG 76317450 IC50 = 1310 nM T16769 C31BXK 76324810 IC50 = 19 nM T16769 CA14LJ 76328363 IC50 = 95 nM T16769 CJ9A3T 76335645 IC50 = 600 nM T16769 C2UVF7 76335647 IC50 = 15 nM T16769 CX0R6S 86276147 IC50 = 4 nM T16769 CZQO17 86650974 IC50 = 320 nM T16769 CBOP84 90089572 IC50 = 100 nM T16769 C73MBT 90089727 IC50 = 45 nM T16769 CO96QE 90089737 IC50 = 40 nM T16769 C10KBD 90231909 IC50 = 220 nM T16769 C3JK9T 90231969 EC50 = 150 nM T16769 COS5A9 90231983 EC50 = 17 nM T16769 CQ5ZA2 90231985 IC50 = 150 nM T16769 C0EMK4 90232067 IC50 = 110 nM T16769 CW98BE 90232119 EC50 = 17 nM T16769 C72DSF 90232137 IC50 = 250 nM T16769 CE6W1R 90232149 EC50 = 13 nM T16769 C75QBJ 90232154 IC50 = 44 nM T16769 C35JLR 90232165 EC50 = 32 nM T16769 CDP7U6 90232174 EC50 = 37 nM T16769 CXI3Y0 90232180 EC50 = 67 nM T16769 CN4D0A 90232202 EC50 = 73 nM T16769 CW74HX 90232234 EC50 = 130 nM T16769 CY0MI8 90232282 EC50 = 180 nM T16769 COQ63T 90232294 IC50 = 13000 nM T16769 C8IQ1M 90232300 EC50 = 69 nM T16769 CN95GA 90232303 EC50 = 14 nM T16769 C4MK9X 90240297 EC50 = 24 nM T16769 C7XF3W 90251750 IC50 = 640 nM T16769 CMU3A7 90654375 IC50 = 2200 nM T16769 CJQ78L 90654376 IC50 = 5200 nM T16769 C6CMZ9 90654377 IC50 = 2500 nM T16769 CY56XM 90654378 IC50 = 3000 nM T16769 CHC78P 90654379 IC50 = 8300 nM T16769 CTHF31 90654380 IC50 > 10000 nM T16769 C6K0WI 90654381 IC50 = 1600 nM T16769 C3HEA9 90654382 IC50 = 3700 nM T16769 CA9HX4 90654383 IC50 = 1300 nM T16769 CN6M3I 90654384 IC50 > 10000 nM T16769 C9K0OL 90654385 IC50 > 10000 nM T16769 CORF34 90654386 IC50 > 10000 nM T16769 CO21FQ 90654387 IC50 > 10000 nM T16769 CP85YF 90654388 IC50 > 10000 nM T16769 CHMQ92 90654389 IC50 > 10000 nM T16769 C72LMU 90654390 IC50 > 10000 nM T16769 CSE3L7 90654391 IC50 > 10000 nM T16769 CJ3Z7O 90654392 IC50 > 10000 nM T16769 CZSK32 90654393 IC50 > 10000 nM T16769 CYM9Z1 90654394 IC50 = 750 nM T16769 COTH12 90654395 IC50 = 940 nM T16769 CG5XS4 90654396 IC50 = 5700 nM T16769 C7GJS1 90654397 IC50 > 10000 nM T16769 C6NW4S 90654398 IC50 = 370 nM T16769 C6YW1O 90654399 IC50 = 1200 nM T16769 CN0V9Q 90654400 IC50 = 6300 nM T16769 C5JLE7 90654401 IC50 = 4800 nM T16769 COR48A 90654402 IC50 = 6700 nM T16769 CIZQ28 90654403 IC50 = 770 nM T16769 CI9Q7H 90654404 IC50 = 990 nM T16769 CSB8J0 90654405 IC50 = 3100 nM T16769 CCQ73R 90654406 IC50 = 1000 nM T16769 CD46OI 90654407 IC50 = 1500 nM T16769 CI23DO 90654408 IC50 = 2000 nM T16769 C1A9HP 90654409 IC50 = 3300 nM T16769 C10DYO 90654410 IC50 = 9200 nM T16769 CM6S3P 90654411 IC50 = 3000 nM T16769 CM59ZC 90654412 IC50 = 1800 nM T16769 CZNT70 90654413 IC50 > 10000 nM T16769 CIH5V8 90664859 IC50 = 2200 nM T16769 CI3MX1 91826683 IC50 = 110000 nM T16769 CA67UG 118323269 IC50 = 58 nM T16769 C0DGE4 118497975 IC50 = 37 nM T16769 C9BSI6 118557690 IC50 = 20 nM T16769 CY82JZ 118557732 IC50 = 14 nM T16769 C6VWZ8 118557745 IC50 = 47 nM T16769 CQ5PB0 118715864 IC50 = 60 nM T16769 CH42OT 118715865 IC50 = 7.9 nM T16769 CDK9H0 118715866 IC50 = 20 nM T16769 C81MSI 118715867 IC50 = 10 nM T16769 C3TGF5 118715868 IC50 = 9.5 nM T16769 CEZ9T6 118715869 IC50 = 3.6 nM T16769 C14FGL 122187534 EC50 = 9.4 nM T16769 CT3OK0 126502413 IC50 = 5.4 nM T16769 C6G3QT 126502414 IC50 = 1.6 nM T16769 C0QVU3 126502417 IC50 = 0.83 nM T16769 COM04R 126502421 IC50 = 14 nM T16769 CM1QX6 132584225 IC50 = 22300 nM T16769 C6NFD0 134419123 IC50 = 94 nM T16769 C6QG3S 137652289 IC50 = 1.4 nM T16769 CL7TG3 137652943 IC50 = 1.7 nM T16769 CUL3H1 137655590 IC50 = 1.1 nM T16769 CXA8J2 137660821 IC50 = 119.3 nM T16769 CK0IX4 137662073 IC50 = 91 nM T16769 C87BOG 138377561 IC50 = 67 nM T16769 C0B8GK 138377594 IC50 = 120 nM T16769 CA43ML 142585287 IC50 = 190.7 nM T16769 CGF6R2 142585309 IC50 = 229.4 nM T16769 C0HC8R 142585337 IC50 = 175.9 nM T16769 C0RHF1 142585361 IC50 > 10000 nM T16769 C5AI8Z 142585365 IC50 = 5944 nM T16769 CM7IG2 142585375 IC50 = 275.7 nM T16769 CG46IU 145954838 IC50 > 1000 nM T16769 CZ25IO 145957358 IC50 = 17 nM T16769 CKEJ30 145979040 IC50 = 16.6 nM T16769 C7XM4Q 145979112 IC50 = 86.8 nM T16769 CWKM51 145979441 IC50 = 8660 nM T16769 CLRM52 145979809 IC50 = 10 nM T16769 CGN1J0 145980475 IC50 = 38.3 nM T16769 CL4F9B 145981512 IC50 = 215.3 nM T16769 CDQ0T6 145981705 IC50 = 15900 nM T16769 C1K6AY 145982930 IC50 = 189.4 nM T16769 C3L1ZW 145985393 IC50 = 76.9 nM T16769 CY8JR0 145986444 IC50 = 35 nM T16769 CE8N3X 145987231 IC50 = 1010 nM T16769 C1HWA3 145988725 IC50 = 47.3 nM T16769 C87AJL 145988932 IC50 = 21900 nM T16769 CVWI49 145990949 IC50 = 4130 nM T16769 CTQ21M 145991361 IC50 = 27300 nM T16769 CX7AV2 145991404 IC50 = 23.2 nM T16769 CPI0F4 145992202 IC50 = 1760 nM T16769 C79EXP 145992527 IC50 = 37.1 nM T16769 CFW27N 145992560 IC50 = 10900 nM T16769 CI4C2R 145992946 IC50 = 6260 nM T16769 C4QID1 145993905 IC50 = 11900 nM T16769 CX1P5T 155261305 IC50 = 65 nM T16769 CZN82L 155512547 IC50 = 4.5 nM T16769 CK8JB2 155512591 IC50 = 28 nM T16769 C4NS5A 155516652 IC50 = 3.5 nM T16769 C0TKW2 155521668 IC50 = 370 nM T16769 CDXW38 155522163 IC50 > 10000 nM T16769 CD38SB 155522648 IC50 > 10000 nM T16769 CEH0W4 155523271 IC50 = 16.6 nM T16769 CI6RN2 155525834 IC50 > 10000 nM T16769 CTVO12 155529198 IC50 = 86 nM T16769 CM4C0S 155530758 IC50 = 85 nM T16769 C0J3ZE 155535472 IC50 = 16 nM T16769 CD54MG 155537330 IC50 = 3.5 nM T16769 C8D7EI 155553655 IC50 = 21 nM T16769 C23UZA 155554597 IC50 = 11 nM T16769 CF3UV1 155556312 IC50 = 1090 nM T16769 CR3UQ4 155561157 IC50 = 12 nM T16769 CH35AZ 155563735 IC50 = 1.4 nM T16769 D03KZH 25172871 Ki = 110.9 nM T16769 D09BKS 44460581 IC50 = 570 nM T16769 D0BW7P 44589292 Ki = 61 nM T16769 D0E7NV 44460469 IC50 = 2800 nM T16769 D0G3TK 5280863 IC50 > 100000 nM T16769 D0Q7TL 24754886 Ki = 26 nM T16769 D0VK7M 49847690 IC50 = 15 nM T83174 D0E3TC 44259 IC50 = 31.6 nM T83174 D03BNU 59604787 IC50 > 10000 nM T83174 D0CV8T 874670 IC50 = 5000 nM T83174 CJ17AM 4877 IC50 > 100000 nM T83174 C8GAZ7 8394 IC50 = 589000 nM T83174 CU2MH3 13623 IC50 = 728000 nM T83174 C38VYU 408991 IC50 = 1570000 nM T83174 C8IOH3 643398 IC50 = 1556000 nM T83174 C4A7CE 737222 IC50 = 37000 nM T83174 CA93IF 2736118 IC50 = 927000 nM T83174 CN6O5K 2769564 IC50 = 1312000 nM T83174 CEJ29F 2779769 IC50 = 1423000 nM T83174 C65MSO 2795564 IC50 = 2216000 nM T83174 CI08MZ 3039701 IC50 = 424000 nM T83174 C70WJL 4679494 IC50 = 1677000 nM T83174 CC8PD6 11389493 IC50 = 1300000 nM T83174 CU0E8O 11690457 Ki > 10000 nM T83174 CB0AP2 11705863 Ki > 10000 nM T83174 C9TU1O 16046126 IC50 > 1000 nM T83174 C0H8UN 16730109 IC50 > 40000 nM T83174 CGP40H 16784276 IC50 = 2000 nM T83174 CIK53Z 22273643 IC50 = 615000 nM T83174 CPSU68 23515094 IC50 > 384000 nM T83174 CSI5Q7 23515103 IC50 = 374000 nM T83174 CTY40O 24229745 IC50 = 229000 nM T83174 C7YG1N 24759534 IC50 = 1500 nM T83174 CX1HL8 25032704 Ki > 8330 nM T83174 CPZ87C 26076409 IC50 = 452000 nM T83174 CLH54Z 29431956 IC50 > 384000 nM T83174 C81QIG 30174069 IC50 = 23000 nM T83174 CLS29B 46872626 IC50 > 10000 nM T83174 CD2K4R 50908681 Ki > 1000000 nM T83174 CM42BY 51000510 Ki > 1000000 nM T83174 CUK1H2 52023984 IC50 > 384000 nM T83174 CWN0L5 57477672 IC50 = 201000 nM T83174 C09SZA 57482985 IC50 = 371000 nM T83174 C9AZ5G 58065595 IC50 = 77000 nM T83174 CXJ63M 59603829 IC50 = 6700 nM T83174 CQEU96 59603842 IC50 = 37 nM T83174 CI7DY2 60965486 IC50 = 900 nM T83174 CLZT12 62059850 IC50 = 22000 nM T83174 C6MV0A 62155416 IC50 > 384000 nM T83174 CV63UL 67240318 IC50 > 10000 nM T83174 C5DGR9 69036886 IC50 = 10000 nM T83174 CX3H4C 71009783 IC50 = 900 nM T83174 C1Q3JE 71062665 IC50 > 384000 nM T83174 C1HW4B 89735655 IC50 = 720 nM T83174 C0KWB7 136525509 IC50 = 34000 nM T83174 CW86XP 138377600 IC50 = 340 nM T83174 C49QOZ 138393053 IC50 = 2.8 nM T83174 C9IY7P 145964008 IC50 = 3.8 nM T83174 C2SVM8 145964907 IC50 = 9500 nM T83174 C8G7QD 145964922 IC50 = 120 nM T83174 C4ZU2L 145965049 IC50 = 110 nM T83174 CDI75R 145965697 IC50 = 148000 nM T83174 CKLJ63 145965749 IC50 = 1100 nM T83174 CIQ70O 145966247 IC50 = 65 nM T83174 CPH9E3 145967023 IC50 = 48 nM T83174 CU3G2V 145967167 IC50 > 384000 nM T83174 CDBG73 145967194 IC50 = 41000 nM T83174 C2TMZ3 145967445 IC50 = 2.7 nM T83174 CX9W8D 145967523 IC50 = 95000 nM T83174 C8CQ2I 145968693 IC50 = 6000 nM T83174 C3PO1Q 145971398 IC50 = 6.5 nM T83174 C32DBK 145971841 IC50 = 7000 nM T83174 CMXU60 145972550 IC50 = 38000 nM T83174 C35ADS 145973250 IC50 = 290 nM T83174 C6EBA0 145973658 IC50 = 7500 nM T83174 CGU24W 145973756 IC50 = 7700 nM T83174 C0O1LK 145974662 IC50 > 384000 nM T83174 C53VBI 145974831 IC50 = 4800 nM T83174 C4FP9E 145975243 IC50 = 30 nM T83174 CMH8Q5 145975400 IC50 = 5 nM T83174 C5FWH2 145975520 IC50 = 105000 nM T83174 CER2C6 145975823 IC50 = 215000 nM T83174 CW62SG 145976074 IC50 = 20000 nM T83174 C5V0AH 145977027 IC50 > 384000 nM T83174 CHSP21 145977039 IC50 = 188000 nM T83174 C1QY5N 145977386 IC50 = 570 nM T83174 C76GEI 145977626 IC50 = 75000 nM T83174 C7MOH6 145978090 IC50 = 800 nM T83174 C78FPU 145978821 IC50 = 221000 nM T83174 C2MD1Q 155513187 IC50 > 10000 nM T83174 C57VPG 155514784 IC50 = 32000 nM T83174 CEL1F7 155514953 IC50 = 710 nM T83174 C14EAF 155518403 IC50 = 76000 nM T83174 CLI4Y7 155521170 IC50 = 263000 nM T83174 CK3HL8 155523714 IC50 > 384000 nM T83174 CL85NA 155541166 IC50 = 270 nM T83174 CC05JX 155542183 IC50 = 19600 nM T83174 CU75ED 155551092 IC50 = 42200 nM T83174 C6JC4W 155553646 IC50 = 24000 nM T83174 COU19A 155555715 IC50 > 384000 nM T83174 D0TO6S 2396 IC50 = 3463 nM T58298 CN5OC4 23673110 Ki = 10700 nM T58298 CZ19JA 24948922 Ki = 161000 nM T58298 CZE07Q 24949080 Ki = 55200 nM T58298 C6IUX2 24949081 Ki = 182000 nM T58298 CLR27K 24949082 Ki = 786000 nM T58298 CVM2K0 24949230 Ki = 154000 nM T58298 C2KS8Z 45141993 IC50 = 20000 nM T58298 CRZ62F 73355036 IC50 = 16100 nM T58298 CDF79W 145950387 IC50 > 300000 nM T58298 C9VIW7 145951405 IC50 > 300000 nM T58298 CI0DE8 145952129 IC50 > 300000 nM T58298 C8WY3S 145952263 IC50 > 300000 nM T58298 CCE24P 145953494 IC50 > 300000 nM T58298 CHSD24 145955401 IC50 > 300000 nM T58298 CVM5E8 145957948 IC50 > 300000 nM T58298 CVC6A1 145958826 IC50 > 300000 nM T58298 C8LWV3 145958854 IC50 > 300000 nM T58298 CYG9B0 145958960 IC50 > 300000 nM T58298 C6YJ4N 145961405 IC50 > 300000 nM T58298 CJ0IQ6 145962930 IC50 > 300000 nM T58298 CHN5E3 145974297 IC50 > 300000 nM T58298 CAU3Z1 146020618 IC50 > 20000 nM T58298 D06GQY 91934096 Ki = 2590 nM T58298 D0DZ1K 45141593 Ki > 40000 nM T28418 D06KTJ 53252276 IC50 = 31 nM T28418 D0E3TC 44259 IC50 = 49.8 nM T28418 D0T3ME 156422 IC50 = 630 nM T28418 CQN3Z7 24825710 IC50 = 686 nM T28418 CCFQ29 44187005 IC50 = 95.3 nM T28418 C8NA4L 53384644 IC50 > 30000 nM T28418 CV63UL 67240318 IC50 > 10000 nM T28418 CPG3A5 86302574 IC50 > 30000 nM T28418 C9WGB8 127035904 IC50 = 3000 nM T28418 CUO0C5 132156633 IC50 > 10000 nM T28418 C2MD1Q 155513187 IC50 > 10000 nM T28418 D05FXD 44478401 IC50 = 2.9 nM T28418 D0X8BU 71718651 IC50 = 2300 nM T71141 D01TJY 53340771 IC50 = 1.4 nM T71141 D09ZXO 176873 IC50 = 10000 nM T71141 CC86KB 492972 Ki = 1.995 nM T71141 CY7WS4 9799158 IC50 = 9600 nM T71141 C68UYS 9808123 IC50 = 1.13 nM T71141 CVTP38 9808486 IC50 = 588 nM T71141 C4LTP2 9825687 IC50 = 754 nM T71141 C13KPA 9848051 Ki < 10000 nM T71141 CB2TS1 9850990 IC50 = 615 nM T71141 CJ7SP4 9851336 IC50 = 52 nM T71141 CTM7V0 9851337 IC50 = 11.7 nM T71141 CVXG48 9862253 IC50 = 4360 nM T71141 C6PNG8 9894403 IC50 = 6000 nM T71141 C2W7NP 9894622 IC50 = 8624 nM T71141 CC6PJ4 9908437 IC50 = 19800 nM T71141 CKRZ62 9937119 IC50 = 64 nM T71141 C9CKS6 9956141 IC50 = 2390 nM T71141 CT4V2Y 9979833 IC50 = 8225 nM T71141 CYA0W2 9983143 IC50 > 10000 nM T71141 C6CWQ8 10003119 IC50 = 5057 nM T71141 CA2SU9 10004734 IC50 = 323 nM T71141 CEJ31C 10027119 IC50 = 2119 nM T71141 CY0T9L 10030149 IC50 > 10000 nM T71141 CLS1F7 10051002 IC50 = 486 nM T71141 COH3U6 10052945 IC50 = 189 nM T71141 CX6H0Q 10072507 IC50 = 164 nM T71141 CK0G2T 10073952 IC50 = 1743 nM T71141 CC3LU6 10074467 IC50 = 25.9 nM T71141 CL47PJ 10096030 IC50 = 216 nM T71141 CLN76R 10096459 IC50 = 0.6 nM T71141 CS2A6F 10098382 IC50 = 352 nM T71141 C4GEW5 10111539 IC50 = 794.33 nM T71141 C1H4NB 10132697 IC50 = 2568 nM T71141 CDL31V 10165701 IC50 = 3730 nM T71141 CO8D9C 10196873 IC50 = 68 nM T71141 C42BVA 10251325 IC50 = 6830 nM T71141 CM9UQ8 10252576 IC50 = 4762 nM T71141 CUZ1I2 10256289 IC50 = 131 nM T71141 C38UIQ 10273975 IC50 = 251.19 nM T71141 CD04QE 10279663 IC50 = 2420 nM T71141 CR2YI9 10297636 IC50 = 674 nM T71141 CX52DZ 10338161 IC50 = 10000 nM T71141 CD1C7I 10345263 IC50 = 3020 nM T71141 CXF75S 10367371 IC50 = 313 nM T71141 CQ04DG 10367832 IC50 = 1433 nM T71141 CL3RB6 10368999 IC50 = 491 nM T71141 C8PNS3 10391689 IC50 = 1394 nM T71141 CC0L8M 10392074 IC50 = 0.04 nM T71141 CEP9G0 10410948 IC50 = 1308 nM T71141 CX1D5C 10411516 IC50 = 350 nM T71141 CB3K1N 10412117 IC50 = 347 nM T71141 CR0F1T 10412890 IC50 = 4623 nM T71141 CUHY62 10433896 IC50 = 2660 nM T71141 CRP82B 10435346 IC50 = 300 nM T71141 C9F2QA 10436174 IC50 = 2671 nM T71141 C1ME0S 10436235 IC50 = 1633 nM T71141 C04HQK 10437073 IC50 = 465 nM T71141 CA27PJ 10478285 IC50 = 66.4 nM T71141 C8EKH9 10479033 IC50 = 1323 nM T71141 C5FX7L 10479186 IC50 = 2444 nM T71141 C0NVB7 10479802 IC50 = 3263 nM T71141 C6IAB4 10482388 IC50 = 4301 nM T71141 C9OM3L 10482416 IC50 = 2108 nM T71141 C6R4MV 10678165 IC50 = 44 nM T71141 C4XFU2 10767331 IC50 = 3800 nM T71141 C08BCF 10993678 IC50 = 4 nM T71141 CDK7W9 10994476 IC50 = 0.4 nM T71141 CTW0P5 11102917 IC50 = 0.15 nM T71141 C79OJR 11133736 IC50 = 61 nM T71141 C5NEM0 11546965 IC50 = 1590 nM T71141 CJ3Q2G 11754575 IC50 = 841 nM T71141 CDVB07 15850631 IC50 = 2000 nM T71141 CG9FV3 15850632 IC50 = 900 nM T71141 CM0JY3 22319462 IC50 = 20000 nM T71141 CGR8U4 22347512 IC50 = 4500 nM T71141 CHP6U7 22347519 IC50 = 10000 nM T71141 CE2G6D 22347593 IC50 = 9800 nM T71141 CIO36K 22347604 IC50 = 4330 nM T71141 CA2C8K 22347617 IC50 = 9600 nM T71141 C5K8AO 22347633 IC50 = 10000 nM T71141 CZ4O2D 44407529 IC50 = 2670 nM T71141 C1E7HF 44407560 IC50 = 4360 nM T71141 C7CP1X 44407779 IC50 = 6240 nM T71141 C5LF3K 44412296 IC50 > 10000 nM T71141 CZ7Q2H 44423872 IC50 = 25000 nM T71141 CKQ84P 44423882 IC50 = 3531 nM T71141 C4R7IN 44429070 IC50 = 3000 nM T71141 CU4ME6 44429074 IC50 = 24 nM T71141 C2XN7B 44429081 IC50 = 20 nM T71141 CZ05RQ 44429084 IC50 = 16 nM T71141 C2EPI3 44429086 IC50 = 42 nM T71141 CHMJ47 44429089 IC50 = 14 nM T71141 CAK98T 44429091 IC50 = 2740 nM T71141 C7J9AT 44429095 IC50 = 6543 nM T71141 C0IUL1 44429100 IC50 = 3532 nM T71141 CC6FH0 44429107 IC50 = 1416 nM T71141 CY1NM2 44429112 IC50 = 366 nM T71141 CE6WM2 44429118 IC50 = 7258 nM T71141 CVW52C 44429121 IC50 = 1835 nM T71141 C0Y9RK 44429125 IC50 = 3443 nM T71141 C7CNA1 44429126 IC50 = 151 nM T71141 C7IO1Q 44429128 IC50 = 88 nM T71141 CW7HB6 44429142 IC50 = 48 nM T71141 C07LGP 44429143 IC50 = 22804 nM T71141 CEW73I 44429144 IC50 = 25 nM T71141 CAX24B 44429145 IC50 = 71 nM T71141 CYV86W 44429146 IC50 = 216 nM T71141 C1PE8W 44429147 IC50 = 96 nM T71141 C8PTR0 44429148 IC50 = 204 nM T71141 CR58CB 44429149 IC50 = 3211 nM T71141 C87WFU 44429150 IC50 = 25 nM T71141 CG6H7J 44429151 IC50 = 1755 nM T71141 C8TNX7 44429152 IC50 = 3420 nM T71141 CD1IN9 44429153 IC50 = 2790 nM T71141 C7MTE0 44429154 IC50 = 1777 nM T71141 CAS34H 44429155 IC50 = 10000 nM T71141 C89OWZ 44429156 IC50 = 631 nM T71141 C4K0NT 44429157 IC50 = 11475 nM T71141 C0C9KL 44429158 IC50 = 622 nM T71141 CVSI23 44429159 IC50 = 12253 nM T71141 CEHF56 44429160 IC50 = 164 nM T71141 C8E3SH 44429161 IC50 = 688 nM T71141 CT47WG 44429162 IC50 = 118 nM T71141 CA01YX 44429163 IC50 = 65 nM T71141 CTM39A 44429164 IC50 = 20 nM T71141 CGQU48 44429165 IC50 = 49 nM T71141 CF5U9Z 44429166 IC50 = 57 nM T71141 COU58G 44429167 IC50 = 40 nM T71141 CN8GI9 44429168 IC50 = 11 nM T71141 CP7U9T 50907449 IC50 = 106 nM T71141 CU65XM 69693295 IC50 = 1258.93 nM T71141 C31IUF 69863577 IC50 = 4 nM T71141 C8EM7Y 71550913 IC50 = 20 nM T71141 CU95LC 71574160 IC50 = 140 nM T71141 COJ8Y4 71574161 IC50 = 19 nM T71141 C8V4UB 71574356 IC50 = 92 nM T71141 CMRQ12 71719408 IC50 = 33 nM T71141 C8B7QE 72949858 IC50 = 1.5 nM T71141 CF1UL2 73348680 IC50 = 2400 nM T71141 CXM8L3 75002097 IC50 = 1995.26 nM T71141 C30NBD 86272865 Ki = 0.01 nM T71141 CW8UV5 86272868 Ki = 0.03981 nM T71141 CCQP95 89979082 IC50 = 200 nM T71141 C2J3VA 118721315 IC50 = 1000 nM T71141 C0BT3F 118721316 IC50 > 10000 nM T71141 C4TNZ0 118721317 IC50 = 398.11 nM T71141 C2N6WI 118721318 IC50 > 10000 nM T71141 CMQ94S 118721319 IC50 = 251.19 nM T71141 C5CW9O 118721320 IC50 = 398.11 nM T71141 CYL2X3 118721321 IC50 = 316.23 nM T71141 CFQA95 118721322 IC50 = 501.19 nM T71141 CWDE71 118721323 IC50 = 398.11 nM T71141 CM9J4X 118721324 IC50 = 794.33 nM T71141 CY13BE 118721325 IC50 = 501.19 nM T71141 C8UNZ5 118721326 IC50 = 398.11 nM T71141 CG5B9F 118721327 IC50 = 630.96 nM T71141 CMXJ63 118721328 IC50 = 630.96 nM T71141 C2OJX9 118721329 IC50 = 630.96 nM T71141 C0YG4M 118721330 IC50 = 398.11 nM T71141 C8F4DG 118721331 IC50 = 251.19 nM T71141 C2ESU9 118721332 IC50 = 100 nM T71141 C2OYU9 118721333 IC50 = 79.43 nM T71141 CX0R3H 118721334 IC50 = 6309.57 nM T71141 CP8I3D 118721335 IC50 = 199.53 nM T71141 CGM28Y 118721336 IC50 = 7943.28 nM T71141 COM73D 118721337 IC50 = 199.53 nM T71141 CH25GR 118721338 IC50 = 158.49 nM T71141 CE7D1S 118721339 IC50 = 199.53 nM T71141 CZ95CL 118721340 IC50 = 158.49 nM T71141 C0AL1C 118721341 IC50 = 501.19 nM T71141 CAZ6U3 118721342 IC50 = 316.23 nM T71141 C65KQW 118721343 IC50 = 63.1 nM T71141 CGJ9O5 118978102 Ki = 0.02512 nM T71141 CL2ER8 121242162 IC50 = 10 nM T71141 CPS9N3 121245322 Ki = 0.07943 nM T71141 C8P7OW 121245346 Ki = 0.03162 nM T71141 CJ83VH 121245350 IC50 = 6309.57 nM T71141 CFOM46 121246727 Ki = 0.03981 nM T71141 CL5Q9G 121246911 IC50 = 1.585 nM T71141 CAL43C 121246982 IC50 = 6.31 nM T71141 C6XK2Y 121247103 IC50 = 2.512 nM T71141 CR5X1T 130453989 Ki = 0.03981 nM T71141 CVT2U3 130454024 IC50 = 2.512 nM T71141 CT4BY6 130454058 IC50 = 1 nM T71141 CZK41V 130454091 Ki = 0.0631 nM T71141 C2OJ3C 130454093 Ki = 0.01995 nM T71141 CU73IM 131985420 IC50 = 1.585 nM T71141 CQEK82 131985476 IC50 = 7.943 nM T71141 C20ZAT 131985489 Ki = 0.03981 nM T71141 C1IKD6 131985494 Ki = 0.05012 nM T71141 CI6W9O 131985523 IC50 = 1.995 nM T71141 C57BQS 132561360 IC50 = 158.49 nM T71141 CXZ16C 137480037 Ki = 0.0631 nM T71141 CV6JY5 139030528 Ki = 0.1072 nM T71141 CAK31T 139593557 IC50 = 15.85 nM T71141 CH9UP3 145982517 IC50 = 12.59 nM T71141 CX0P5N 145982847 Ki = 0.07943 nM T71141 CL13NC 145982905 Ki = 0.1 nM T71141 C4N5TW 145983050 Ki = 0.0631 nM T71141 CJ70YV 145984499 Ki = 0.07943 nM T71141 C4R5NQ 145984560 IC50 = 39.81 nM T71141 CM9FS1 145985439 IC50 = 50.12 nM T71141 CRA6D0 145985939 IC50 = 3.981 nM T71141 CB2X7V 155511318 IC50 = 398.11 nM T71141 COVD01 155511742 IC50 = 204 nM T71141 C2MG6X 155512266 IC50 = 40.7 nM T71141 CJ41WG 155514043 IC50 = 460 nM T71141 C7LI4B 155514586 IC50 = 630.96 nM T71141 CSMQ36 155514765 IC50 = 251.19 nM T71141 CHT1J6 155515540 IC50 = 0.26 nM T71141 CQ5C4M 155516533 IC50 = 47 nM T71141 CAOY19 155516610 IC50 = 31.62 nM T71141 CO9F1P 155517149 IC50 = 707 nM T71141 CB8HQ4 155518124 IC50 = 73 nM T71141 CE1D6N 155518125 IC50 = 12.59 nM T71141 C4RBX6 155518148 IC50 = 42.4 nM T71141 C35OHK 155518750 IC50 = 1.995 nM T71141 CTA5S4 155518784 IC50 = 12.59 nM T71141 CT5I4G 155519672 IC50 = 769 nM T71141 CPD07V 155519834 IC50 = 14.5 nM T71141 C6BPT7 155520545 IC50 = 31.8 nM T71141 CMF13G 155520959 IC50 = 63.1 nM T71141 CL5K1Z 155521171 IC50 = 316.23 nM T71141 CL7OU0 155521485 IC50 = 100 nM T71141 C5WQV7 155522262 IC50 = 69.9 nM T71141 C52NID 155522392 IC50 = 70 nM T71141 C9OR7L 155522422 IC50 = 1000 nM T71141 CEL76H 155523874 IC50 = 29.6 nM T71141 CB6WM8 155524349 IC50 = 114 nM T71141 C0NJ9Y 155526007 IC50 = 264 nM T71141 C90YTQ 155526362 IC50 = 79.43 nM T71141 CC2QW3 155526724 IC50 = 62 nM T71141 CZ68AU 155528189 IC50 = 19.95 nM T71141 CG1TX8 155530618 IC50 = 95 nM T71141 C6LAW0 155533172 IC50 = 125.89 nM T71141 CN5DO1 155533902 IC50 = 215 nM T71141 C56FZV 155534494 IC50 = 180 nM T71141 CJ7O2X 155534687 IC50 = 99 nM T71141 C3QT6L 155534872 IC50 = 794.33 nM T71141 CW9MN7 155535114 IC50 = 889 nM T71141 CS03LO 155538904 IC50 = 6.31 nM T71141 C1ELZ5 155539211 IC50 = 223 nM T71141 CB2S3T 155539763 IC50 = 94.5 nM T71141 CAH63Q 155540069 IC50 = 48.4 nM T71141 CR36QP 155540115 IC50 = 39.81 nM T71141 CE1W5B 155540544 IC50 = 19498.45 nM T71141 CYW32T 155541264 IC50 = 79.43 nM T71141 CN1AH9 155542562 IC50 = 40.2 nM T71141 CX49AZ 155542672 IC50 = 274 nM T71141 CJ89TS 155543010 IC50 = 13.4 nM T71141 CJC2T1 155545083 IC50 = 559 nM T71141 CFGD59 155545309 IC50 = 1554 nM T71141 CB96AH 155545672 IC50 = 50.12 nM T71141 CHO8K7 155546051 IC50 = 139 nM T71141 COP7I6 155546233 IC50 = 8.3 nM T71141 C7QO1R 155547533 IC50 = 142 nM T71141 CZGB26 155547699 IC50 = 39 nM T71141 C38CME 155548638 IC50 = 187 nM T71141 C10EIB 155549200 IC50 = 74 nM T71141 CLW19Y 155549414 IC50 = 369 nM T71141 CLN24G 155549618 IC50 = 826 nM T71141 CJZ35U 155549685 IC50 = 25.12 nM T71141 CC95ZO 155551413 IC50 = 256 nM T71141 CWF98D 155552156 IC50 = 160 nM T71141 C89SLB 155552170 IC50 = 223 nM T71141 CW5AV4 155552698 IC50 = 158.49 nM T71141 C1D8GP 155553166 IC50 = 495 nM T71141 C2SRV6 155553944 IC50 = 75.9 nM T71141 CV4DG6 155554134 IC50 = 31.62 nM T71141 C29DNJ 155554489 IC50 = 31 nM T71141 C0BDS6 155556102 IC50 = 720 nM T71141 C2F1UL 155557078 IC50 = 449 nM T71141 C2VIB1 155557895 IC50 = 112.4 nM T71141 C08HEW 155560738 IC50 = 417 nM T71141 C4U2RS 155563179 IC50 = 324 nM T71141 CKRE58 155563328 Ki = 0.1738 nM T71141 C35CXQ 155563458 IC50 = 140 nM T71141 CR50VG 155563627 IC50 = 420 nM T71141 CEF3T8 155563936 IC50 = 0.67 nM T71141 C3FL5Z 155565918 IC50 = 430 nM T71141 CP2D3H 155566033 IC50 = 81.3 nM T71141 C5GQX9 155567527 IC50 = 39.81 nM T71141 C1HNT9 155567705 IC50 = 12.59 nM T71141 CYZ02H 155568897 IC50 = 12589.25 nM T71141 C7Z4RD 155569291 IC50 = 7.943 nM T39797 CCI84V 155511169 IC50 = 4.8 nM T39797 C1Y5KS 155513541 IC50 = 7.3 nM T39797 CBU43W 155522465 IC50 = 9.2 nM T39797 C59ERX 155554358 IC50 = 53 nM T39797 CA5XJ8 155556372 IC50 = 32 nM T84160 D0H3HM 60795 Ki = 501.19 nM T84160 D0K0KH 656665 Ki = 5.3 nM T84160 D0K7WK 4595 Ki = 7.6 nM T84160 D0R1JV 60854 Ki = 398.11 nM T84160 D0R6RO 4184 IC50 = 1412.54 nM T84160 D0S9MU 5078 IC50 > 10000 nM T84160 D0T8GD 89594 Ki = 71000 nM T84160 D0V4QS 135398745 Ki = 199.53 nM T84160 D0Z1RV 135398737 Ki = 398.11 nM T84160 D0Z6UC 5358 IC50 > 10000 nM T84160 D00OWF 5280953 Ki > 10000 nM T84160 D06DZI 107780 Ki = 6309.57 nM T84160 D0S6PJ 5012 Ki = 58 nM T84160 D0V3GT 671690 IC50 = 9.3 nM T84160 D0ZG9N 132337 Ki = 152 nM T84160 D0ZX7I 131747 Ki = 103 nM T84160 C5JG6U 2689 IC50 = 1318.26 nM T84160 CZUI83 2769 Ki = 152 nM T84160 CTO54F 4442 Ki = 0.071 nM T84160 C5FJD1 10832 Ki > 10000 nM T84160 C28OSR 14623 Ki = 12 nM T84160 C1MK7I 16075 Ki > 10000 nM T84160 C0YU1V 16157 Ki = 2340 nM T84160 C9F3EI 19933 Ki = 200 nM T84160 CF4WA9 20882 Ki = 220 nM T84160 C9ZO6A 21527 Ki = 725 nM T84160 CX4TB5 29667 Ki = 780 nM T84160 C2MO8K 29669 Ki = 62 nM T84160 C2A3IV 41357 Ki = 1200 nM T84160 CN6RO2 69747 Ki > 10000 nM T84160 CZ6G7B 69873 Ki > 10000 nM T84160 C3JXH7 97478 Ki = 2160 nM T84160 CKP25M 121881 Ki = 199.53 nM T84160 CLP01Z 139381 Ki > 10000 nM T84160 C2VPW8 151947 Ki = 12 nM T84160 CGT8R0 160510 Ki > 10000 nM T84160 C8YMA9 176469 Ki > 10000 nM T84160 C10TAR 182588 Ki = 0.47 nM T84160 CLH68M 228022 Ki = 6520 nM T84160 C39OMI 269722 Ki = 1640 nM T84160 CX0M5S 316974 Ki > 10000 nM T84160 CH6BG7 376254 EC50 = 3 nM T84160 CU4O0N 407233 Ki > 10000 nM T84160 C32CWP 409364 Ki = 442 nM T84160 C40FKT 409370 Ki = 18 nM T84160 CYV1R3 417052 Ki > 10000 nM T84160 CV8ZW5 504350 Ki = 1460 nM T84160 CC6Y2H 2730263 Ki = 890 nM T84160 C37EYD 2730269 Ki = 225 nM T84160 CW68MS 2730436 Ki > 10000 nM T84160 CYR1J2 2735754 Ki = 40 nM T84160 CR40QK 2736204 Ki > 10000 nM T84160 C4ZUJ5 2757788 Ki = 320 nM T84160 CY4MH1 3024499 Ki = 15 nM T84160 C3W2DI 3057577 Ki = 1250 nM T84160 CPKW92 3073104 Ki = 1.5 nM T84160 CBJ03H 3073168 Ki = 6.1 nM T84160 CJ40RA 3596754 EC50 = 7.2 nM T84160 CB49JS 3613700 Ki = 3.1 nM T84160 CIR7L6 3621644 Ki = 990 nM T84160 CXFS34 3835333 Ki = 126 nM T84160 C1VS4C 4203196 Ki = 243 nM T84160 CY7PH0 4302960 Ki < 10000 nM T84160 CXG39N 4327008 EC50 = 15 nM T84160 CHF96N 5173985 Ki = 2440 nM T84160 C9O3LP 7018035 Ki = 1600 nM T84160 C8P7LB 9572056 Ki > 10000 nM T84160 C6YDQ0 9795278 Ki = 1662 nM T84160 C6I4QG 9841032 IC50 = 0.0008128 nM T84160 CFI97S 9904205 IC50 = 1202.26 nM T84160 C9B3EA 9911844 Ki < 1000 nM T84160 CA17GY 9922799 Ki = 2024 nM T84160 C0C7NV 9930121 Ki = 511 nM T84160 COD73F 9943346 Ki = 580 nM T84160 C7TS9J 9944605 Ki = 409 nM T84160 CIWG38 10015966 Ki = 1.1 nM T84160 CGRX96 10035245 Ki = 34 nM T84160 C2JZL1 10048222 IC50 > 1000 nM T84160 C7O5DA 10061682 Ki = 10 nM T84160 CUW74G 10064052 IC50 > 1000 nM T84160 CM4T5H 10243306 Ki = 0.7 nM T84160 CVF1E5 10246054 IC50 > 1000 nM T84160 CSE47M 10247171 IC50 = 4.571 nM T84160 CNJ03F 10374840 Ki = 32 nM T84160 C78PBC 10378253 Ki = 0.23 nM T84160 CDAC63 10381889 IC50 = 478.63 nM T84160 C58GMP 10419235 Ki = 2910 nM T84160 C4S5NL 10423801 EC50 = 3.8 nM T84160 CLDM93 10445840 Ki = 310 nM T84160 CG16KL 10447948 Ki = 0.83 nM T84160 C94TVH 10452995 IC50 = 6.607 nM T84160 C3IY9P 10498554 IC50 = 3019.95 nM T84160 CTP65K 10519608 IC50 = 45.71 nM T84160 CH1ZM2 10521333 EC50 = 4.2 nM T84160 CP8NL9 10521792 Ki = 420 nM T84160 CX18VH 10522259 EC50 = 12 nM T84160 CZ2H5B 10543269 EC50 = 54 nM T84160 CFN8B5 10546440 IC50 = 2.399 nM T84160 C1LV7P 10548259 IC50 = 0.7943 nM T84160 CE59TG 10553922 IC50 = 87.1 nM T84160 CART26 10569395 IC50 = 19.5 nM T84160 C9GSI8 10571450 IC50 = 13.49 nM T84160 CF19LK 10583272 Ki > 10000 nM T84160 C7WP3H 10587905 EC50 = 2.7 nM T84160 C5WA7Q 10594684 EC50 = 4.2 nM T84160 CRY9Q0 10617292 IC50 = 0.3548 nM T84160 C39FNQ 10619583 IC50 = 20.42 nM T84160 C86KEZ 10620679 IC50 = 19.5 nM T84160 C7DQP5 10632134 Ki > 10000 nM T84160 C01MLV 10637485 IC50 = 0.003981 nM T84160 CCS31Z 10645335 IC50 = 1288.25 nM T84160 CV3LH2 10655071 Ki > 10000 nM T84160 CQIG19 10655345 Ki = 560 nM T84160 C07AKO 10663820 IC50 = 28183.83 nM T84160 C4PV2W 10666301 IC50 = 2.63 nM T84160 CB3C9Z 10667071 IC50 = 14.13 nM T84160 C54PZD 10667842 Ki > 10000 nM T84160 CB52LK 10679485 Ki > 10000 nM T84160 C8T4WH 10683189 EC50 = 9.5 nM T84160 CC54NZ 10707897 EC50 = 14 nM T84160 CD7ZW9 10712829 EC50 = 6.6 nM T84160 C9FAP1 10714457 IC50 = 2570.4 nM T84160 CIBU90 10714509 IC50 > 100000 nM T84160 CVS29F 10715484 IC50 = 117.49 nM T84160 CB49LK 10726651 Ki > 10000 nM T84160 CPH26L 10727230 Ki = 38 nM T84160 CY1M6L 10738329 IC50 = 0.2884 nM T84160 CNB5C6 10750797 Ki = 660 nM T84160 CZO1E3 10753377 IC50 = 1.479 nM T84160 C17OFU 10756517 IC50 = 0.912 nM T84160 CQK9U8 10778246 EC50 = 1.7 nM T84160 CY0D7K 10804369 Ki = 48 nM T84160 CZ73FW 10805206 EC50 = 2.4 nM T84160 C8S4PF 10808909 IC50 = 1.175 nM T84160 CB1W8Z 10826756 EC50 = 1.6 nM T84160 C0JPR3 10831864 Ki = 1450 nM T84160 CL0BO9 10834414 IC50 = 30.9 nM T84160 CBD60Q 10853821 IC50 = 27542.29 nM T84160 CYG3H9 11543786 Ki = 174 nM T84160 CQ2Z8J 11738788 Ki = 2225 nM T84160 CPG15O 11743399 IC50 > 1000 nM T84160 C90MLE 11797241 IC50 = 28.18 nM T84160 C1M3BY 11797762 IC50 = 37153.52 nM T84160 CXLW54 11948707 Ki > 10000 nM T84160 CB34AR 11957729 Ki = 7.2 nM T84160 CC09BF 12118765 Ki > 10000 nM T84160 CZ15UV 12253678 Ki = 190 nM T84160 C51RAV 12253688 Ki = 5 nM T84160 CN0B8T 12253699 Ki = 2710 nM T84160 CHNE61 12253771 Ki > 10000 nM T84160 C04VGK 12996853 Ki > 10000 nM T84160 C8SG1D 13041565 Ki > 10000 nM T84160 CMTC02 14639161 Ki > 10000 nM T84160 CK21HZ 15226949 IC50 = 12.02 nM T84160 CM5Z8L 15595236 Ki > 10000 nM T84160 C5E0JF 17221604 Ki = 1200 nM T84160 COF61U 17982621 Ki = 49.8 nM T84160 C7UAD4 18950026 Ki = 274 nM T84160 C6AOE8 19426635 IC50 > 1000 nM T84160 CQ7WI4 19689601 Ki = 450 nM T84160 C74ESH 19793429 Ki = 60 nM T84160 CPRB74 19793437 Ki = 0.68 nM T84160 CJ30MF 19793443 Ki = 63 nM T84160 C6MRH5 19793461 Ki = 67 nM T84160 CK71LJ 19841587 Ki = 230 nM T84160 CQ3JL0 19956256 IC50 = 120.23 nM T84160 CLVT08 19978038 IC50 = 0.9772 nM T84160 CF34NC 19978059 IC50 = 0.08128 nM T84160 C60FRA 20543488 Ki = 6200 nM T84160 C1L5IR 21680423 Ki = 38 nM T84160 CQY54O 22246875 Ki > 10000 nM T84160 C90DNQ 23599502 Ki = 1547 nM T84160 C9MR6L 44269164 Ki = 2.7 nM T84160 CKX4C3 44286463 Ki = 0.23 nM T84160 CKWM20 44287807 Ki = 40 nM T84160 CG5NY0 44287946 Ki > 10000 nM T84160 C1XN0G 44288126 Ki = 36 nM T84160 C1IWT4 44296810 IC50 > 100000 nM T84160 C8MY6X 44305741 Ki = 44.67 nM T84160 CN27ME 44305742 Ki = 20.42 nM T84160 CYKA50 44305829 Ki = 14.45 nM T84160 CP3K1N 44305830 Ki = 1.38 nM T84160 C9ZO0B 44305831 Ki = 28.18 nM T84160 CZP31C 44305849 Ki = 40.74 nM T84160 CV8WZ0 44318454 IC50 > 1000 nM T84160 CXJL56 44318842 IC50 > 1000 nM T84160 CEH42A 44322540 Ki = 690 nM T84160 C2RO6E 44325521 Ki = 0.51 nM T84160 C98WVB 44339912 Ki = 0.86 nM T84160 CY5DC6 44339913 Ki = 0.39 nM T84160 C2Y0LH 44339926 Ki = 19 nM T84160 CNDH74 44339931 Ki = 42 nM T84160 C3VKD6 44339932 Ki = 3.2 nM T84160 CPX9B7 44339933 Ki = 0.44 nM T84160 C3J0KC 44339934 Ki = 0.88 nM T84160 CM1Z5Y 44339938 Ki = 71 nM T84160 CL4QW0 44339942 Ki = 53 nM T84160 CV6WF1 44339951 Ki = 0.58 nM T84160 CBU80G 44339954 Ki = 0.51 nM T84160 CU0P6N 44339976 Ki = 1.3 nM T84160 C6O2MU 44340011 Ki = 1.1 nM T84160 CM0P8C 44340023 Ki = 0.45 nM T84160 C9U7KH 44340030 Ki = 0.32 nM T84160 C5L8GJ 44340073 Ki = 2.6 nM T84160 C97LDQ 44340205 Ki = 0.96 nM T84160 C8WI0A 44340224 Ki = 1.1 nM T84160 CETW50 44340225 Ki = 1.5 nM T84160 CZYX47 44340582 Ki = 0.69 nM T84160 CJGD80 44340583 Ki = 7.2 nM T84160 CA30OX 44343077 Ki = 9 nM T84160 C46VYW 44352664 Ki > 10000 nM T84160 C7K6ER 44352705 Ki = 150 nM T84160 CS1H8C 44360164 IC50 = 6.918 nM T84160 C8MLC3 44360191 IC50 = 28.84 nM T84160 C1F7SQ 44360192 IC50 = 1.995 nM T84160 C4GW7P 44360218 IC50 = 23.44 nM T84160 C3XEC1 44360645 IC50 = 218.78 nM T84160 CNZE83 44360648 IC50 = 5.754 nM T84160 C06XBQ 44360649 IC50 = 2.512 nM T84160 CCEN16 44360668 IC50 = 87.1 nM T84160 C3XF2K 44360669 IC50 = 33.88 nM T84160 CJ5MP3 44360695 IC50 = 1.995 nM T84160 C6UCQ7 44360696 IC50 = 218.78 nM T84160 C5AOP4 44360709 IC50 = 14.13 nM T84160 C1L5JK 44360710 IC50 = 3.981 nM T84160 C3MDJ1 44360711 IC50 = 3.467 nM T84160 C4IU6A 44360712 IC50 = 5.012 nM T84160 CGS8M7 44360732 IC50 = 23.99 nM T84160 CG5JN2 44360760 IC50 = 288.4 nM T84160 C3C2TD 44402933 Ki = 665 nM T84160 C1APT8 44402939 Ki = 1043 nM T84160 CG87PW 44409290 Ki > 1000 nM T84160 C74FIE 54681508 Ki = 1.4 nM T84160 CHR72D 54681510 Ki = 6.4 nM T84160 C0CZ8R 54681514 Ki = 0.48 nM T84160 CDI84E 71450922 IC50 = 10 nM T84160 CP9TR0 10324985 Ki > 10000 nM T84160 D01KAX 135453290 Ki > 10000 nM T84160 D03TDN 1342 Ki = 175 nM T84160 D04AXY 9993659 Ki = 1.9 nM T84160 D05GDP 599482 Ki > 10000 nM T84160 D08BCF 5011 IC50 = 0.4467 nM T84160 D09RPR 16737207 Ki > 10000 nM T84160 D0C9TY 16727408 Ki = 73 nM T84160 D0F6CD 5202 Ki = 120 nM T84160 D0G2BS 5013 Ki = 3 nM T84160 D0H4NK 4780 Ki = 1200 nM T84160 D0J6JT 1355 Ki = 62 nM T84160 D0M5ZE 5311416 Ki = 501.19 nM T84160 D0P2HR 3510 Ki = 2.1 nM T84160 D0R9AD 558969 Ki = 1.8 nM T84160 D0S0XK 9863146 IC50 = 1.413 nM T84160 D0SA4A 1354 Ki = 17 nM T84160 D0T3QZ 5311136 Ki = 1.622 nM T84160 D0V4RP 1346 Ki = 2500 nM T84160 D0V5HV 4296 Ki = 1390 nM T84160 D0W2YN 2760172 Ki = 32 nM T84160 D0X4RC 7096 Ki = 3000 nM T84397 CX42YI 23757 IC50 = 4800 nM T84397 CS8H7I 55708 IC50 = 1500 nM T84397 CM47KI 5351344 IC50 = 180 nM T84397 C1LS0K 5386397 IC50 = 33000 nM T84397 C4CFR8 5466706 IC50 = 3400 nM T84397 C7N8QY 6439188 IC50 = 10000 nM T84397 CVT2F0 6473980 IC50 = 2500 nM T84397 CB51HV 9884538 IC50 = 620 nM T84397 C0PNJ2 10066775 IC50 = 3310 nM T84397 CRL1B9 10110183 IC50 = 2400 nM T84397 CTB37M 10150010 IC50 = 450 nM T84397 CE1DG7 10154653 IC50 = 1200 nM T84397 CDQ05P 10155421 IC50 = 650 nM T84397 CJTZ14 10155655 IC50 = 12000 nM T84397 C6KCY3 10157011 IC50 > 10000 nM T84397 CJ97VC 10157446 IC50 = 1700 nM T84397 C2WCI1 10193563 IC50 = 7900 nM T84397 C2V6TC 10193933 IC50 = 470 nM T84397 CVD8L5 10215598 IC50 = 4000 nM T84397 CFA01X 10215648 IC50 = 31000 nM T84397 C7LP0A 10215785 IC50 = 510 nM T84397 CTU3A1 10286758 IC50 = 2000 nM T84397 CY5AQ2 10309096 IC50 > 10000 nM T84397 C2M6WY 10336128 IC50 = 7200 nM T84397 C9VP5G 10359957 IC50 = 2180 nM T84397 C18JWT 10380369 IC50 > 100000 nM T84397 CT6LY7 10405034 IC50 = 3760 nM T84397 CU8M6G 10451021 IC50 = 460 nM T84397 CB2Q4Y 10473384 IC50 = 900 nM T84397 CQT8O9 10617491 IC50 = 2600 nM T84397 CXO5K4 10880163 IC50 = 700 nM T84397 CL53UK 10880474 IC50 = 4500 nM T84397 C4RC1W 10881066 IC50 = 2000 nM T84397 C4ZQU9 10901245 IC50 = 6600 nM T84397 CLT14P 10915864 IC50 = 1100 nM T84397 C8UIK9 10915865 IC50 = 31000 nM T84397 CA7Y4E 11035782 IC50 = 1200 nM T84397 C7IKJ4 11064916 IC50 = 650 nM T84397 CD5AF7 11107890 IC50 = 3100 nM T84397 CRL3E9 11142886 IC50 = 500 nM T84397 C20KVY 11157967 IC50 = 3800 nM T84397 CC3DR0 11162707 IC50 = 2690 nM T84397 C4XEW2 11164846 IC50 > 40000 nM T84397 CK9Q5G 11187974 IC50 = 6500 nM T84397 C1L5OA 11259802 IC50 > 40000 nM T84397 C39UJV 11316806 IC50 = 7600 nM T84397 C90LVO 11335997 IC50 = 1300 nM T84397 C9F0OU 11340271 IC50 > 40000 nM T84397 C91WOY 11341288 IC50 > 40000 nM T84397 C5N4OU 11352927 IC50 > 40000 nM T84397 CM1G7E 11359891 IC50 = 130 nM T84397 C7HP6L 11371837 IC50 = 2800 nM T84397 CXC86U 11373611 IC50 > 40000 nM T84397 C28NCQ 11396761 IC50 > 40000 nM T84397 C9PIN3 11438919 IC50 = 130 nM T84397 C50HXY 11442353 IC50 > 40000 nM T84397 CVK7B8 11453615 IC50 = 20000 nM T84397 C9JK3P 11460836 IC50 = 14000 nM T84397 C5U3NZ 11750977 IC50 > 40000 nM T84397 C7ECZ9 11777823 IC50 = 120 nM T84397 C62GWL 11780979 IC50 = 5500 nM T84397 CF2UK7 14977376 IC50 > 100000 nM T84397 COEV92 44367259 IC50 = 560 nM T84397 C2I3WS 44367274 IC50 = 21000 nM T84397 C7BS5H 44367323 IC50 > 100000 nM T84397 C1S2BL 44367324 IC50 > 100000 nM T84397 CWH0N9 44367333 IC50 = 41000 nM T84397 C60AMC 44392097 IC50 = 13000 nM T84397 CSQB32 44400801 IC50 = 1250 nM T84397 CSI58X 44400846 IC50 = 9000 nM T84397 C5SN6P 44400896 IC50 > 100000 nM T84397 D01DMN 234105 IC50 = 2900 nM T84397 D04XJT 44367275 IC50 = 11000 nM T84397 D0LH3S 5388779 IC50 = 200 nM T01575 D07UHS 107970 IC50 = 17000 nM T01575 D09ZWH 135564845 IC50 > 100000 nM T01575 C5UGO6 25066518 IC50 > 30000 nM T01575 CAU96H 44186115 IC50 > 30000 nM T01575 CM8H5Z 44186480 IC50 = 2400 nM T01575 CX7J6K 59240661 IC50 = 3400 nM T01575 C7E3RN 90644083 IC50 = 30000 nM T01575 C0RHZ2 90644084 IC50 = 740 nM T01575 CCS21I 90644085 IC50 > 30000 nM T01575 CA0YP4 90644086 IC50 = 1700 nM T01575 C4KV8N 90644087 IC50 = 2500 nM T01575 CH1OL9 90644088 IC50 > 30000 nM T01575 CV3N9P 90644089 IC50 > 30000 nM T01575 C92VMG 90644090 IC50 > 30000 nM T01575 CG6X9K 90644091 IC50 = 30000 nM T01575 C3D4OP 90644092 IC50 = 2300 nM T01575 CX71RE 90644093 IC50 = 12000 nM T01575 CWQ10N 90644094 IC50 = 100 nM T01575 CQ3H6T 90644095 IC50 = 1300 nM T01575 CFHB98 90644096 IC50 = 24 nM T01575 CMB3U1 118796836 IC50 = 485 nM T01575 CNA52R 127045779 IC50 = 39200 nM T01575 C1JI8T 127046000 IC50 = 9600 nM T01575 CZ4T2K 127046001 IC50 = 150 nM T01575 CSH59B 127046002 IC50 = 150 nM T01575 CAU6F5 127046003 IC50 = 1000 nM T01575 C5HTI9 127046004 IC50 = 117 nM T01575 CL32ZV 127046006 IC50 = 1000 nM T01575 C68XAU 127046007 IC50 = 3800 nM T01575 C2V8TU 127046008 IC50 = 9200 nM T01575 C29KUT 127046212 IC50 = 930 nM T01575 C2IU0Y 127046404 IC50 = 4600 nM T01575 CNYM51 127046405 IC50 = 590 nM T01575 C0C7PM 127046409 IC50 = 730 nM T01575 C8VMH6 127046410 IC50 = 50000 nM T01575 CH39AZ 127046411 IC50 = 7300 nM T01575 CA1CR7 127046569 IC50 = 5000 nM T01575 C1VAS8 127046570 IC50 = 25000 nM T01575 CR0AF5 127046571 IC50 > 50000 nM T01575 CET21P 127046603 IC50 = 6400 nM T01575 C8FO1I 127047987 IC50 = 1200 nM T01575 CV7N0S 127047998 IC50 = 720 nM T01575 D0K4YP 108037 IC50 > 100000 nM T01575 D0S5OU 73729049 IC50 = 210 nM T93903 D0J3SU 9847835 Ki = 120 nM T93903 C1RUH9 4246483 IC50 = 93000 nM T93903 CO58XD 5311161 IC50 > 100000 nM T93903 CFN2P6 9800285 Ki = 850 nM T93903 CLTO67 9821317 IC50 = 5 nM T93903 C4XO3K 9821545 Ki = 1200 nM T93903 CJI5T3 9823027 IC50 = 160 nM T93903 C74QTI 9823074 IC50 = 2720 nM T93903 C6S3KT 9840223 Ki = 1100 nM T93903 CD05OL 9867192 IC50 = 230 nM T93903 CX67SZ 10826725 Ki = 5000 nM T93903 CPM09W 11166638 EC50 = 290 nM T93903 CM8O6L 11257152 IC50 = 30 nM T93903 CCV6T0 11374367 IC50 = 9 nM T93903 CD8WB9 44304162 Ki > 50000 nM T93903 CXR1V5 44434249 IC50 = 6 nM T93903 CGY3W2 71471109 IC50 = 1000 nM T93903 CANH70 71716242 IC50 = 1100 nM T93903 C40WIR 71718085 IC50 = 1740 nM T93903 CU75VK 71719897 IC50 = 800 nM T93903 CBV6F1 71720507 IC50 = 2300 nM T93903 CQ9H4U 86277844 IC50 = 5000 nM T93903 C9QKI3 127020966 IC50 > 100000 nM T93903 C73BEC 155527521 EC50 = 310 nM T93903 CD7ZU4 155528030 EC50 = 240 nM T93903 CU42CE 155567829 IC50 > 100000 nM T93903 D0N5MU 4117381 Ki = 12000 nM T93903 D0Q9XX 515950 Ki = 7200 nM T93903 D0Y5IQ 44255320 IC50 = 5000 nM T40111 D06IAR 60961 Ki > 100000 nM T40111 CSR10C 510912 IC50 = 55 nM T40111 COJ29X 890649 IC50 = 5600 nM T40111 C7TZ5D 2930546 IC50 = 20300 nM T40111 C70OXL 3006288 Ki = 15400 nM T40111 CF8N3B 3140491 EC50 > 50000 nM T40111 CAY86S 3312427 IC50 = 8600 nM T40111 CIXQ25 6478685 IC50 = 1500 nM T40111 CW62YA 6479888 IC50 = 770 nM T40111 CN29OD 6618978 IC50 > 50000 nM T40111 CLIF21 9842306 IC50 = 38 nM T40111 CM73SE 9858793 IC50 = 46 nM T40111 CGB78L 9880305 IC50 = 55 nM T40111 CW3S9G 9883477 IC50 = 99 nM T40111 CG16TY 9907596 IC50 = 160 nM T40111 C2X6TP 10233633 Ki = 520 nM T40111 C05NVJ 10259194 Ki = 300 nM T40111 CGF36N 10315709 IC50 = 90 nM T40111 C71JXF 10652408 Ki = 260 nM T40111 CLYM27 10746991 Ki = 340 nM T40111 CDT59Z 10841975 Ki = 37970 nM T40111 CT8DX2 11069304 Ki = 890 nM T40111 C17DLS 11828231 Ki = 2300 nM T40111 C54TFI 12093480 IC50 > 1000 nM T40111 C34QTH 15625173 IC50 = 2600 nM T40111 C3DLS6 15625174 IC50 = 3100 nM T40111 CYX2U3 15625175 IC50 = 1100 nM T40111 CD8B6T 15625184 IC50 = 10900 nM T40111 CJI3P1 15625185 IC50 = 22700 nM T40111 C4X0BA 15625186 IC50 = 2600 nM T40111 CESJ49 15625187 IC50 = 2500 nM T40111 CFLV58 15625188 IC50 = 1800 nM T40111 CX1DZ0 15625192 IC50 = 1200 nM T40111 C8FP9H 15625193 IC50 = 940 nM T40111 CP3L1T 15625194 IC50 = 1800 nM T40111 C1N8XS 16007061 IC50 = 37 nM T40111 C4RKU7 16046198 Ki = 20 nM T40111 CKTA70 16484765 IC50 = 6300 nM T40111 CH0R7U 16484780 IC50 = 9900 nM T40111 CN5AB6 16747704 Ki = 23600 nM T40111 CS42ZC 23626089 IC50 = 4100 nM T40111 CJO79M 23644735 Ki = 73 nM T40111 C2NW5X 23648220 Ki = 19 nM T40111 CCN63I 23648221 Ki = 20 nM T40111 CMVH63 23648222 Ki = 7 nM T40111 C0OR1M 23648223 Ki = 45 nM T40111 C5PIF4 23648224 Ki = 45 nM T40111 C90FQM 23648225 Ki = 10 nM T40111 CB35PV 23648226 Ki = 96 nM T40111 CQ90NK 23648227 Ki = 1 nM T40111 CKZT87 23648228 Ki = 66 nM T40111 CBC71W 23648229 Ki = 16 nM T40111 CYG18K 24748985 Ki = 2070 nM T40111 C6M4QN 24748986 Ki = 5000 nM T40111 CK32AR 24749071 Ki = 400 nM T40111 C9E0AU 24749072 Ki = 2830 nM T40111 CO6DB0 25147739 Ki = 350 nM T40111 C09KIE 25181866 Ki = 7800 nM T40111 CND10S 25181867 Ki > 100000 nM T40111 CX5BU0 25181868 Ki = 2300 nM T40111 C68PMG 25181869 Ki = 44000 nM T40111 C5JVN4 25210968 Ki = 20800 nM T40111 CUZT43 25210969 Ki = 10300 nM T40111 CW8I0P 25879063 IC50 = 150 nM T40111 CXM9L0 44367538 IC50 = 150 nM T40111 CZID50 44367579 IC50 = 83 nM T40111 C70YFO 44415246 Ki = 87 nM T40111 CRZW96 44415248 Ki = 20 nM T40111 C16EMS 44433349 IC50 = 67000 nM T40111 CC2UO4 44440695 IC50 = 23600 nM T40111 COQ83H 44578784 IC50 = 23600 nM T40111 C84EYU 44578785 Ki = 660 nM T40111 C8GJB9 44578786 Ki = 520 nM T40111 C9T2EI 44578787 Ki = 820 nM T40111 CIK76G 44578789 Ki > 100000 nM T40111 CEI32X 44589747 Ki = 42800 nM T40111 C2MF0S 44589785 Ki > 100000 nM T40111 CG7WJ4 44589786 Ki = 97300 nM T40111 CVO20H 46839190 Ki = 14000 nM T40111 C3GET9 46839191 Ki = 77 nM T40111 C0SV8O 46839192 Ki = 1500 nM T40111 C1V3CQ 46839320 Ki = 70 nM T40111 C01DSF 46876831 Ki = 660 nM T40111 CG3RM9 46876832 Ki = 330 nM T40111 CIT31Y 46927861 Ki = 300 nM T40111 CXW02B 46927862 Ki = 580 nM T40111 CU4Z3R 49864088 Ki = 17000 nM T40111 CP5HR1 49864089 Ki = 4400 nM T40111 CQ39WM 49864090 Ki = 1200 nM T40111 C76JYP 49864102 Ki = 8200 nM T40111 CN2G3Z 49864103 Ki = 7100 nM T40111 C01GAC 49864104 Ki = 460 nM T40111 CR8E0Z 51351534 Ki = 5 nM T40111 C9YL2W 51351535 Ki = 99 nM T40111 CPY1M0 51351558 Ki = 16 nM T40111 CT64YQ 52905544 Ki = 522 nM T40111 C81NCO 53317433 Ki = 1100 nM T40111 C81TOB 53317434 Ki = 349 nM T40111 C7R4DT 53317435 Ki = 255 nM T40111 CZ4FR9 53317436 Ki = 77 nM T40111 C0MC6P 53320028 Ki = 5550 nM T40111 C64FAH 53320029 Ki = 14200 nM T40111 CQU37F 53320030 Ki = 94 nM T40111 CFO5E7 53320031 Ki = 70 nM T40111 CN32LO 53320311 Ki = 95 nM T40111 CPO0F3 53322659 Ki = 87 nM T40111 CMT39Y 53322660 Ki = 7900 nM T40111 CN6Q8M 53324226 Ki = 1 nM T40111 CC9D8J 53326788 Ki = 13 nM T40111 C39KQY 71716568 Ki = 110 nM T40111 C3M0JK 72163956 IC50 = 105 nM T40111 CNQ2D6 72945146 Ki = 491 nM T40111 C5OJ0X 72945148 Ki = 39 nM T40111 C01HVL 72945149 Ki = 163 nM T40111 C1OVC0 72945150 Ki = 2553 nM T40111 CBPC50 72945349 Ki = 265 nM T40111 C7MJQ5 72945350 Ki = 3771 nM T40111 C9NTH1 72945351 Ki = 132 nM T40111 CVJ0N8 72945352 Ki = 19 nM T40111 CP1I9N 72945353 Ki = 7723 nM T40111 CJ4R8C 72945541 Ki = 2035 nM T40111 C74WCI 72945542 Ki = 3 nM T40111 C7T3HN 72945732 Ki = 5.6 nM T40111 C95BZQ 72947911 Ki = 13 nM T40111 CCVO01 72947912 Ki = 0.6 nM T40111 CB7HG8 72948102 Ki = 63 nM T40111 C4U3OA 72948103 Ki = 82 nM T40111 CX2U3L 72948104 Ki = 70 nM T40111 C3N7OD 72948105 Ki = 876 nM T40111 CZJ5F6 73346517 Ki = 5556 nM T40111 CN5QE0 73346518 Ki = 892 nM T40111 C26EXZ 73349141 IC50 = 558 nM T40111 CAD90T 73349545 Ki = 4362 nM T40111 CD4BY1 73351103 Ki = 4308 nM T40111 CB94EM 73352218 IC50 = 680 nM T40111 CWO9Q0 73352572 Ki = 854 nM T40111 CPS4I8 76309998 Ki = 38 nM T40111 CB2PT6 76309999 Ki = 56 nM T40111 CL42ER 76310000 Ki = 1679 nM T40111 CI1J4W 76310001 Ki = 1017 nM T40111 CEB47C 76310002 Ki = 2811 nM T40111 C3ICR7 76310003 Ki = 906 nM T40111 C7C9FJ 76317234 Ki = 56 nM T40111 CTLJ38 76317235 Ki = 1828 nM T40111 CZ9U2T 76320941 Ki = 733 nM T40111 C7HJC1 76324606 Ki = 259 nM T40111 C0DFQ1 76328163 Ki = 144 nM T40111 CL41TU 76328164 Ki = 5127 nM T40111 C86TRQ 76331843 Ki = 32 nM T40111 CTFG08 76331844 Ki = 2203 nM T40111 C3OVW6 76335415 Ki = 164 nM T40111 CG7Z4S 76335416 Ki = 259 nM T40111 CD9S8B 90663694 Ki = 110 nM T40111 C1GPY5 145952889 IC50 = 11100 nM T40111 CFQ2O9 145954131 IC50 > 30000 nM T40111 C93AKF 145980356 IC50 = 10100 nM T40111 C67YXK 145980711 IC50 = 13200 nM T40111 CWC78S 145983656 IC50 = 4300 nM T40111 C6VP2S 145985880 IC50 > 30000 nM T40111 C5QBJ2 145989469 IC50 = 20400 nM T40111 C20PUW 145990385 IC50 = 7600 nM T40111 CBL59V 145990969 IC50 = 13800 nM T40111 CP42FJ 145991406 IC50 = 7200 nM T40111 D01LDQ 24749070 Ki = 70 nM T40111 D03HDS 6475540 Ki = 520 nM T40111 D07HZQ 444451 Ki = 33 nM T40111 D0A4AL 477579 Ki = 300 nM T40111 D0S4BK 73680 Ki = 100 nM T40111 D0T4UE 44578788 Ki = 18200 nM T40111 D0Z8EV 446541 IC50 = 19 nM T62460 D03ZBT 11626560 IC50 = 563 nM T62460 D04LKS 25126798 Ki = 0.09 nM T62460 D04LVK 57379345 IC50 = 3730 nM T62460 D0EG1I 9926791 IC50 = 0.5 nM T62460 D0Y7IC 44205240 IC50 = 0.99 nM T62460 D00RYA 16750271 IC50 = 2700 nM T62460 D02TUL 118115473 IC50 = 1640 nM T62460 D03HUX 49792852 IC50 > 10000 nM T62460 D03LWG 53235510 IC50 > 10000 nM T62460 D04QWQ 59422203 IC50 = 13.2 nM T62460 D05PCM 78323835 IC50 = 29 nM T62460 D06EIC 57928403 IC50 = 3.9 nM T62460 D07EHV 44814409 IC50 > 10000 nM T62460 D07HPJ 11476171 IC50 > 10000 nM T62460 D07JAG 58557659 IC50 = 8 nM T62460 D0BI3N 44595079 IC50 = 12 nM T62460 D0D5ZJ 25062766 IC50 = 11 nM T62460 D0D8KQ 25127112 IC50 = 10 nM T62460 D0DK5X 135567296 IC50 = 2.2 nM T62460 D0DK8X 50922691 IC50 = 75 nM T62460 D0E3TC 44259 IC50 = 0.627 nM T62460 D0G8BM 16722836 IC50 = 100 nM T62460 D0O0LS 25141092 IC50 = 112 nM T62460 D0PN8H 46216796 IC50 = 1280 nM T62460 D0S1XX 134821691 IC50 = 1 nM T62460 D0SG7B 49831257 IC50 = 10 nM T62460 D0GZ7B 5328779 IC50 = 3380 nM T62460 C1BE5N 3799 IC50 = 19952.62 nM T62460 CU68FI 78893 Ki > 3500 nM T62460 CV7W4J 176406 IC50 = 39810.72 nM T62460 C6ZB4U 790291 Ki = 4600 nM T62460 CGQM48 869412 Ki = 2100 nM T62460 C0XL5P 951379 Ki > 3500 nM T62460 C7ZUW6 1246120 Ki = 3100 nM T62460 CI1B7L 1247281 Ki > 3500 nM T62460 CP6BI3 1481965 IC50 = 30000 nM T62460 C3F0GS 3120536 Ki = 2200 nM T62460 CD67OL 4250390 Ki > 3500 nM T62460 C6SNL5 4393251 Ki > 3500 nM T62460 CG9RD4 4448318 IC50 = 8530 nM T62460 CK6L3O 5121684 Ki > 3500 nM T62460 CYA76E 9798589 IC50 > 100000 nM T62460 CRZ5T7 9815801 IC50 > 10000 nM T62460 CO70CQ 10107882 IC50 = 290 nM T62460 CP28QI 10154513 IC50 > 10000 nM T62460 C35JMD 10269598 IC50 = 1550 nM T62460 C7SFI1 10296883 IC50 = 7300 nM T62460 CK2RY9 11164105 IC50 = 1480 nM T62460 C58YUH 11993785 IC50 = 47 nM T62460 C0Y7MG 12083227 IC50 = 1700 nM T62460 CZI64D 12083230 IC50 = 670 nM T62460 C75SGK 12997800 IC50 = 2 nM T62460 C0DUA7 15953425 IC50 = 14 nM T62460 C3JWA6 15953427 IC50 = 18 nM T62460 CWZM24 15953526 IC50 = 16 nM T62460 C1U8XW 16109036 IC50 = 1300 nM T62460 CSE35D 16739464 IC50 = 1800 nM T62460 C20OFQ 16739508 IC50 = 650 nM T62460 CCP56J 16739905 IC50 = 200 nM T62460 CQ64XI 16739921 IC50 = 390 nM T62460 CM3UF8 16739935 IC50 = 3200 nM T62460 CFEP56 16739948 IC50 = 170 nM T62460 C23KZR 16739951 IC50 > 10000 nM T62460 C9OQ1G 16750272 IC50 = 8000 nM T62460 CW2SY5 16750291 IC50 = 420 nM T62460 CIX7U2 16750304 IC50 = 3000 nM T62460 C6A3XS 16750306 IC50 = 1500 nM T62460 CB2TK1 16750327 IC50 = 1900 nM T62460 CH4O1C 16750328 IC50 > 10000 nM T62460 C90MJD 16750331 IC50 > 10000 nM T62460 C7JW2E 18008439 IC50 > 10000 nM T62460 C6UAZ0 20820292 IC50 = 230 nM T62460 C87BYV 22282847 IC50 > 10000 nM T62460 CJ5GR1 22282945 IC50 > 7140 nM T62460 C50FBN 22282953 IC50 > 10000 nM T62460 C16TAZ 22484511 IC50 = 720 nM T62460 CE7K3W 23532567 IC50 > 10000 nM T62460 CUY98W 23585560 IC50 = 39 nM T62460 CD0R9O 24699546 Ki > 3500 nM T62460 C7YG1N 24759534 IC50 = 2300 nM T62460 CAJ4T2 24762205 IC50 > 10000 nM T62460 CQNP54 24764449 IC50 = 25000 nM T62460 CRO97A 24798484 IC50 = 184 nM T62460 CFS2M7 24798487 IC50 = 142 nM T62460 CLBP72 24798571 IC50 = 70 nM T62460 CX1U4S 24800423 IC50 = 710 nM T62460 C4T0DG 24800602 IC50 = 8900 nM T62460 CH3ZG7 24800604 IC50 = 5300 nM T62460 CBA02Y 24800776 IC50 = 210 nM T62460 C3UFG1 24801129 IC50 = 47 nM T62460 CVR8S1 24801650 IC50 = 760 nM T62460 CWV98O 24899557 IC50 = 1000 nM T62460 C5S7XA 24958852 IC50 = 58 nM T62460 CJ68PR 24958855 IC50 = 180 nM T62460 C0JYA9 25123154 IC50 = 390 nM T62460 C56JVD 25123155 IC50 = 91 nM T62460 CZM6Q2 25123472 IC50 = 35 nM T62460 C3IA7V 25123474 IC50 = 1500 nM T62460 C6V4NB 25123475 IC50 = 460 nM T62460 CFK89A 25123806 IC50 = 98 nM T62460 C3RMN9 25123807 IC50 = 250 nM T62460 C5GO3T 25123808 IC50 = 1850 nM T62460 C4WFL0 25128110 IC50 = 130 nM T62460 COV8Z0 25143021 IC50 > 10000 nM T62460 CI0E2L 25154395 IC50 = 970 nM T62460 CL1W5D 25154436 IC50 = 390 nM T62460 C0ZXH7 25236808 Ki = 1700 nM T62460 CT7X8Y 27700054 Ki > 3500 nM T62460 C9M1PO 42599880 IC50 = 547 nM T62460 C93PID 42599883 IC50 > 10000 nM T62460 CB9DS2 42600632 IC50 = 975 nM T62460 CIA57B 42600635 IC50 = 27 nM T62460 CH10ZY 42600886 IC50 > 10000 nM T62460 C3IT9C 42600887 IC50 > 4000 nM T62460 CY4LG8 42622934 IC50 = 1.5 nM T62460 CCB1E9 44124695 IC50 > 100000 nM T62460 CIT2A7 44192904 IC50 = 256.7 nM T62460 C3VRO9 44557921 IC50 = 4365.16 nM T62460 C5YL2S 44570390 IC50 = 490 nM T62460 C7DW0O 44602589 IC50 = 2.8 nM T62460 C6QT0J 44622837 IC50 > 1000 nM T62460 C4EBH7 44625519 IC50 > 4000 nM T62460 C02RNS 44625983 IC50 = 103 nM T62460 CKUA84 44626045 IC50 = 92 nM T62460 C7E1DT 44626178 IC50 = 23 nM T62460 C2SLI6 44631938 IC50 = 10 nM T62460 CU3RF1 45139989 IC50 > 10000 nM T62460 CQGZ06 45139991 IC50 > 10000 nM T62460 CZ7T8F 45275363 IC50 = 16 nM T62460 CB58EO 45275368 IC50 = 24 nM T62460 CU3AD0 45275473 IC50 = 28 nM T62460 CQ3KO2 45375955 IC50 = 58 nM T62460 CE45XW 46208354 IC50 = 2.9 nM T62460 CUHB49 46208355 IC50 = 2.5 nM T62460 CW38GO 46208357 IC50 = 3.5 nM T62460 C43COY 46208358 IC50 = 5.4 nM T62460 CE4Q7D 46208596 IC50 = 6.7 nM T62460 CM9UN7 46208601 IC50 = 0.24 nM T62460 CH7JB4 46209051 IC50 = 4.2 nM T62460 C7ON5A 46233287 IC50 > 10000 nM T62460 CWN3M0 46234565 IC50 = 92 nM T62460 CLTU68 46234566 IC50 = 26 nM T62460 C5YH1F 46235625 IC50 = 59 nM T62460 CC25DT 46235942 IC50 = 30 nM T62460 CZ7J6K 46236109 IC50 = 83 nM T62460 C1S4LH 46398810 IC50 = 303 nM T62460 C35AIH 46865430 IC50 = 48 nM T62460 C2EK4B 46865431 IC50 = 140 nM T62460 CMZ0R3 46865529 IC50 = 28 nM T62460 C3B2NL 46865530 IC50 = 82 nM T62460 CC2O9R 46865656 IC50 = 1584.89 nM T62460 CJ3NV8 46865657 IC50 = 130 nM T62460 C5NZ8R 46880686 IC50 = 680 nM T62460 CZ79VE 46880687 IC50 = 27.5 nM T62460 C0YNH6 46880737 IC50 = 22 nM T62460 CGO7C5 46880738 IC50 = 82 nM T62460 C75ZTG 46880739 IC50 = 180 nM T62460 C9T7WL 46880784 IC50 = 67 nM T62460 CSV4G2 46880785 IC50 = 35 nM T62460 C9MW2L 46885052 IC50 > 10000 nM T62460 C69HUW 46885053 IC50 = 940 nM T62460 CASL67 46885231 IC50 = 1200 nM T62460 CEU6O4 46885232 IC50 = 4700 nM T62460 CE27LI 46885233 IC50 = 89 nM T62460 CB8LN4 46885234 IC50 = 362 nM T62460 CMX7U6 46885289 IC50 = 190 nM T62460 CB1ZN5 46885290 IC50 = 60 nM T62460 C2B5XF 49765254 IC50 > 10000 nM T62460 CT7EY8 49817363 IC50 = 253 nM T62460 CMKB24 49838268 IC50 = 22 nM T62460 CB34CO 49839441 Ki = 360 nM T62460 C2DGY0 49839445 Ki > 3500 nM T62460 C06MKW 49839561 Ki = 83.8 nM T62460 CJZ5A0 49840306 IC50 > 10000 nM T62460 CF91RS 49843531 IC50 > 10000 nM T62460 C7A6IZ 49850211 IC50 = 20 nM T62460 C9UZ6E 49855558 IC50 > 10000 nM T62460 CR6Q5Y 49855559 IC50 = 1760 nM T62460 CTM0I6 49855750 IC50 = 1200 nM T62460 CJXR91 49855751 IC50 = 2240 nM T62460 C57FQH 49856318 IC50 = 2780 nM T62460 C70QSD 49856319 IC50 = 1120 nM T62460 C24SMN 49856320 IC50 > 10000 nM T62460 CHK7D3 49856321 IC50 = 840 nM T62460 C90VXM 49856700 IC50 = 1910 nM T62460 CK4LJ5 49856703 Ki = 610 nM T62460 CK5TH3 50906783 IC50 = 10 nM T62460 CA0WR3 50914031 IC50 = 170 nM T62460 CQE9D1 50925411 IC50 = 311 nM T62460 C2Y6QS 50938552 IC50 > 10000 nM T62460 CF26MU 50991562 IC50 = 6000 nM T62460 C20VEP 50994284 IC50 > 10000 nM T62460 CI1L0M 50994285 IC50 = 737 nM T62460 C7ZWT8 50994286 IC50 = 4700 nM T62460 C6VNE1 50994366 IC50 = 754 nM T62460 CSEZ73 50994367 IC50 = 6500 nM T62460 C1R8ZI 50995341 IC50 = 509 nM T62460 C53NRD 50995522 IC50 = 621 nM T62460 C9NYP4 51036677 IC50 > 10000 nM T62460 C4WRY3 51037112 IC50 > 10000 nM T62460 CRI28Z 51037948 IC50 > 10000 nM T62460 CA9DE6 52941228 IC50 = 500 nM T62460 C1T5EH 52942437 IC50 = 610 nM T62460 CEPS91 52943663 IC50 = 39 nM T62460 C2IQ5B 52943672 IC50 >= 10000 nM T62460 CTN0C3 52944839 IC50 = 990 nM T62460 CT2U3E 52947304 IC50 = 19 nM T62460 CQY9D0 52948526 IC50 = 45 nM T62460 C8TC3P 52948550 IC50 = 80 nM T62460 CIM43G 52948562 IC50 = 160 nM T62460 CL14DA 53317826 IC50 = 490 nM T62460 C72DMQ 53320251 IC50 > 7500 nM T62460 C2W9OA 53324451 IC50 > 10000 nM T62460 C0PLX8 53340959 Ki = 2.9 nM T62460 CN70RK 53341007 Ki = 9.1 nM T62460 CQS1R8 53341008 Ki = 16 nM T62460 CKS8G7 53341054 Ki = 9.3 nM T62460 CSUN84 53341057 Ki = 14 nM T62460 C4R2SW 53341104 Ki = 2.6 nM T62460 C4BM5W 53341107 Ki = 6.2 nM T62460 CZKQ72 53341161 Ki = 7.9 nM T62460 CN59SH 53341248 Ki = 2.4 nM T62460 CB83XH 53341368 Ki = 24 nM T62460 CD2CH6 53341413 Ki = 25 nM T62460 CGP23R 53341457 Ki = 0.4 nM T62460 CK7O6Y 53341461 Ki = 16 nM T62460 C9QEA5 53341463 Ki = 1.7 nM T62460 C7U1KW 53341498 Ki = 4.6 nM T62460 C5ZI7P 53341503 Ki = 0.9 nM T62460 C2MAO8 53341544 Ki = 22 nM T62460 C56TYK 53385837 IC50 = 430.5 nM T62460 CNLM53 53385838 IC50 = 361 nM T62460 C1XE2K 53385938 IC50 = 870.7 nM T62460 C37JTE 53385939 IC50 = 47 nM T62460 CV92IB 53386254 IC50 = 23 nM T62460 CU6QF7 53386309 IC50 < 0.5 nM T62460 CYU0R4 53386418 IC50 = 0.59 nM T62460 C7RM6Q 53386421 IC50 = 0.47 nM T62460 CEN91X 53389820 IC50 = 636.6 nM T62460 C37PHN 53497571 IC50 = 211 nM T62460 CCF1B3 53497572 IC50 = 1090 nM T62460 CY5C8A 54589404 IC50 = 3.2 nM T62460 CS7E0A 54672927 IC50 = 224.3 nM T62460 CHZ27O 54673255 IC50 = 24 nM T62460 C7X5ZM 54673258 IC50 = 75.8 nM T62460 CZ84NW 54673259 IC50 = 44.5 nM T62460 CX0U2A 54673422 IC50 = 44.8 nM T62460 C19FZK 54673425 IC50 = 1102.5 nM T62460 CBPT15 54673763 IC50 = 6300 nM T62460 C36BAI 54673911 IC50 = 108.1 nM T62460 CD8ZK6 54674056 IC50 = 220 nM T62460 CFTE97 54674369 IC50 = 840 nM T62460 CUCI05 54674990 IC50 = 99.7 nM T62460 CH0IM9 54754557 IC50 = 54 nM T62460 C1XS2J 54760383 IC50 = 3300 nM T62460 CXH2P4 54766274 IC50 = 370 nM T62460 CD28VZ 54766423 IC50 > 10000 nM T62460 CAP1J7 54766425 IC50 > 10000 nM T62460 C75JFM 54766426 IC50 > 10000 nM T62460 CDIC43 54766427 IC50 = 850 nM T62460 C2XDG1 54766428 IC50 = 5400 nM T62460 C0XCY1 54766576 IC50 = 2100 nM T62460 CPH3Y7 54766578 IC50 > 10000 nM T62460 C0T4SL 54766726 IC50 = 480 nM T62460 CZD70Q 54767039 IC50 = 74 nM T62460 CN1DZ6 54767189 IC50 = 150 nM T62460 C1W3EZ 56591424 IC50 = 3.5 nM T62460 CTB63S 56591428 IC50 = 79 nM T62460 CWR1P6 56591446 IC50 = 18 nM T62460 C6ZL7H 56592816 IC50 = 1200 nM T62460 C6Z1QA 56592817 IC50 = 24 nM T62460 CM8JX1 56604907 IC50 = 10000 nM T62460 CR9A5O 56834874 IC50 = 708 nM T62460 C58MSV 56834889 IC50 = 177 nM T62460 CBFR12 56925356 IC50 = 133 nM T62460 C80DRA 56925357 IC50 = 406 nM T62460 C0HUN8 56925358 IC50 = 307 nM T62460 C6Z2EA 56925359 IC50 = 8820 nM T62460 CC1MN2 56925454 IC50 = 3100 nM T62460 C3XC0T 56925455 IC50 = 377 nM T62460 CBW6T3 56925456 IC50 = 39 nM T62460 C8G3NO 56925457 IC50 = 70 nM T62460 CHS19C 56925458 IC50 = 36 nM T62460 CBMO42 56925459 IC50 = 78 nM T62460 CQTD41 56925550 IC50 = 129 nM T62460 CI9T3S 56925551 IC50 = 654 nM T62460 CS84ZU 56925552 IC50 = 206 nM T62460 C9IVD0 56929216 Ki = 1.8 nM T62460 CQ2F3C 56973424 Ki = 1.7 nM T62460 CSO40C 56973425 Ki = 2.4 nM T62460 CU5BD9 57336812 IC50 = 81 nM T62460 C31LJU 57339437 Ki = 10 nM T62460 CMF7J0 57339438 Ki = 45 nM T62460 CPO2J4 57342178 IC50 = 4800 nM T62460 CA93PN 57342180 IC50 = 5100 nM T62460 C9Z6QJ 57502388 IC50 = 43 nM T62460 COU4M1 57915982 IC50 = 20 nM T62460 C1G5SK 57916044 IC50 = 30 nM T62460 C3C0PQ 57916049 IC50 = 79 nM T62460 CH6RB0 57916164 IC50 = 24 nM T62460 C9MF8U 57928260 IC50 = 19 nM T62460 C3KQJ8 57928435 IC50 = 3.9 nM T62460 C5H8VE 57928583 IC50 = 12 nM T62460 C13VIO 57928632 IC50 = 110 nM T62460 C8BTO7 57928826 IC50 = 7.8 nM T62460 C8R4FE 57991377 IC50 = 134.3 nM T62460 CD6ZP3 58009815 EC50 = 430 nM T62460 CWU1Y3 58009825 EC50 = 1200 nM T62460 C8S6MY 58010054 IC50 = 3 nM T62460 CM1B4V 58010265 EC50 = 150 nM T62460 CQND09 58177229 IC50 = 231 nM T62460 CU4I8X 58177247 IC50 = 53 nM T62460 CLEH36 58177279 IC50 = 287 nM T62460 CIK3U8 58177332 IC50 = 129 nM T62460 C8D2TA 58177362 IC50 = 199 nM T62460 CYC85B 58177456 IC50 = 15 nM T62460 C7BU0H 58180518 IC50 = 22 nM T62460 CKA28H 58180521 IC50 = 16 nM T62460 C2I5LO 58180525 IC50 = 61 nM T62460 CN4OZ8 58180573 IC50 = 250 nM T62460 C92FOB 58180591 IC50 = 19 nM T62460 CWXC70 58180596 IC50 = 270 nM T62460 C9N1QB 58180623 IC50 = 330 nM T62460 CSK1U8 58180628 IC50 = 40 nM T62460 C6LT9S 58180630 IC50 = 46 nM T62460 CCBT87 58180639 IC50 = 40 nM T62460 C3MK9V 58374721 IC50 = 1.4 nM T62460 C7Q8YZ 58374808 IC50 = 2749 nM T62460 CP81TW 58394456 Ki = 62 nM T62460 C4H3FY 58394522 Ki = 1.6 nM T62460 CM6SK2 58394565 Ki = 12 nM T62460 C8NFX5 58394608 Ki = 19 nM T62460 C6HPO3 58394632 Ki = 8.5 nM T62460 CBJ47W 58394678 Ki = 96 nM T62460 CC05OW 58394694 Ki = 32 nM T62460 CK71MA 58394722 Ki = 150 nM T62460 C6A8NR 58394745 Ki = 1.2 nM T62460 CH4F5Y 58394751 Ki = 2 nM T62460 C0F3BO 58394783 Ki = 2.8 nM T62460 CLA74K 58394787 Ki = 4.9 nM T62460 C0Y6FH 58394796 Ki = 68 nM T62460 CO5TH6 58394820 Ki = 88 nM T62460 CY0UV6 58394828 Ki = 1.3 nM T62460 C0X7IK 58394837 Ki = 0.9 nM T62460 CW7D0O 58394866 Ki = 0.8 nM T62460 C0W2AT 58394878 Ki = 210 nM T62460 C97QAK 58394904 Ki = 5.8 nM T62460 C9Q4WD 58394916 Ki = 15 nM T62460 CI37CQ 58394927 Ki = 1.3 nM T62460 CFQW46 58394944 Ki = 2.9 nM T62460 C5RGU7 58394946 Ki = 121 nM T62460 CDP7J2 58394959 Ki = 4.3 nM T62460 CF8G9P 58394966 Ki = 50 nM T62460 C6KO0G 58395044 IC50 = 30 nM T62460 CASI81 58395078 Ki = 0.1 nM T62460 C2H4NS 58395107 Ki = 3.7 nM T62460 C3Y6WA 58395132 Ki = 9.3 nM T62460 CCK96S 58395150 Ki = 2.7 nM T62460 CTF2Z1 58395158 Ki = 2.6 nM T62460 C0GSU3 58395193 Ki = 13 nM T62460 CDK5L1 58395223 Ki = 1.5 nM T62460 CU04YA 58395228 Ki = 8.7 nM T62460 CWOB94 58395230 Ki = 0.6 nM T62460 C9J5UV 58395232 Ki = 2 nM T62460 CO7G2W 58395250 Ki = 7.3 nM T62460 C21OFZ 58395252 Ki = 8.3 nM T62460 CYC87B 58395253 Ki = 156 nM T62460 CQP86B 58395268 Ki = 28 nM T62460 CI7KN3 58395278 Ki = 5.8 nM T62460 CTX12W 58395280 Ki = 11 nM T62460 CWBM72 58395283 Ki = 0.3 nM T62460 CA8LU4 58395286 Ki = 5 nM T62460 C5S8BK 58395290 Ki = 18 nM T62460 CCHV76 58395300 Ki = 9.6 nM T62460 C4H2ZP 58395301 Ki = 1.1 nM T62460 CUS1M8 58395328 Ki = 43 nM T62460 C0WBQ9 58395366 Ki = 15 nM T62460 CWO4X6 58395380 Ki = 5.2 nM T62460 C1YJ3U 58395383 Ki = 12 nM T62460 CGV59X 58395401 Ki = 0.6 nM T62460 C8KQE6 58395411 Ki = 18 nM T62460 CWR1A7 58395421 Ki = 3.7 nM T62460 C28ADB 58395446 Ki = 0.9 nM T62460 CZR91G 58395466 Ki = 2.1 nM T62460 CLA5V3 58395468 Ki = 21 nM T62460 C0X5CV 58395476 Ki = 2.1 nM T62460 CR9T7W 58438557 IC50 = 44.7 nM T62460 CY3W6B 58438580 IC50 = 272 nM T62460 CR7C4V 58438607 IC50 = 7.4 nM T62460 C9MIL7 58450666 IC50 = 219 nM T62460 CWX4G9 58522116 IC50 = 5090 nM T62460 C4A6LT 58522124 IC50 = 4390 nM T62460 CI9VB0 58522237 IC50 = 3320 nM T62460 C1LE9A 58522238 IC50 = 3470 nM T62460 C74ACR 58522276 IC50 = 8220 nM T62460 CI0L1J 58522322 IC50 = 4160 nM T62460 CVMO97 58522377 IC50 = 3190 nM T62460 C7S1PR 58522381 IC50 = 2150 nM T62460 C8X6YE 58557497 IC50 = 40 nM T62460 C2GO4H 59186418 IC50 = 3055 nM T62460 CPWM60 59291925 IC50 = 22 nM T62460 CE6KO4 59291951 IC50 = 27 nM T62460 CT3EW2 59292007 IC50 = 4.1 nM T62460 C2PE0T 59292008 IC50 = 35 nM T62460 CU3W2S 59292043 IC50 = 50 nM T62460 CC6J4I 59363349 IC50 = 35 nM T62460 CQ93TM 59363383 IC50 = 15 nM T62460 CKQ31B 59363409 IC50 = 42 nM T62460 CW76YC 59589542 IC50 = 1979 nM T62460 C0DV7R 59589757 IC50 = 156 nM T62460 CM50TL 59589801 IC50 > 10000 nM T62460 CZ0LA4 59589877 IC50 = 418 nM T62460 CXJ63M 59603829 IC50 = 4200 nM T62460 CQEU96 59603842 IC50 = 220 nM T62460 C8UMJ2 59617909 Ki > 3500 nM T62460 CDMO01 59617921 Ki > 3500 nM T62460 CUNY05 59617942 Ki = 1700 nM T62460 CY7V3I 59617971 Ki > 3500 nM T62460 CM6B3E 59618010 Ki > 3500 nM T62460 CQCG48 59618036 Ki > 3500 nM T62460 CJ5GF1 59618081 Ki > 3500 nM T62460 CT12JO 59618117 Ki > 3500 nM T62460 C42OZL 59618123 Ki = 490 nM T62460 COI26N 59618146 Ki > 3500 nM T62460 CR5GJ4 59618147 Ki > 3500 nM T62460 C9GB1C 59618160 Ki > 3500 nM T62460 CR9F7D 59618164 Ki = 2900 nM T62460 C7XWE2 59618171 Ki = 1500 nM T62460 C2EIA3 59618285 Ki = 1000 nM T62460 C1ZKR9 59618313 Ki > 3500 nM T62460 C26BNV 59618424 Ki > 3500 nM T62460 C3B7CU 59618428 Ki = 1000 nM T62460 CBH83T 59618445 Ki = 100 nM T62460 C3HC4P 59618462 Ki > 3500 nM T62460 CX0FQ2 59618505 Ki = 200 nM T62460 CG8ET4 59618513 Ki = 2400 nM T62460 CR27IT 59618564 Ki > 3500 nM T62460 CNY59P 60165955 Ki = 0.5 nM T62460 CY3QT8 60165956 Ki = 12 nM T62460 C9PH1Z 60166106 Ki = 50 nM T62460 CR9J1T 60166239 Ki = 11 nM T62460 CO1K2C 60166359 Ki = 33 nM T62460 CEL3B4 60166360 Ki = 6.1 nM T62460 C9IHN3 60166488 Ki = 4.5 nM T62460 C75BLR 60166489 Ki = 5.9 nM T62460 C4FL2P 60166490 Ki = 2.7 nM T62460 C97PZW 60166491 Ki = 9.5 nM T62460 CYK50X 60166623 Ki = 3.2 nM T62460 CKT4Y7 60170769 Ki = 1.2 nM T62460 C3YSV5 60170770 Ki = 9.3 nM T62460 C34RVN 60170771 Ki = 1.5 nM T62460 C74FPI 60170772 Ki = 4.5 nM T62460 CTC8E4 60170773 Ki = 6.1 nM T62460 CR80CH 60170858 Ki = 2.6 nM T62460 C3PA9G 60170859 Ki = 7.3 nM T62460 C2AEG3 60170860 Ki = 90 nM T62460 CHJM71 60170861 Ki = 4.8 nM T62460 CBP48G 60170862 Ki = 5.4 nM T62460 C3R0NO 63107904 IC50 = 24100 nM T62460 CSZ6I5 66556035 IC50 = 501.19 nM T62460 C7MD5X 66556536 IC50 = 1995.26 nM T62460 CNDH38 66557868 Ki = 0.2 nM T62460 CJ08ZL 66604045 IC50 = 49 nM T62460 CY0I2V 66604274 IC50 = 141 nM T62460 CD0LJ6 66604359 IC50 = 52 nM T62460 CS8HK2 66604394 IC50 = 18 nM T62460 C7U8GC 66604464 IC50 = 67 nM T62460 CXU94O 66604576 IC50 = 169 nM T62460 CE9T0V 66604664 IC50 = 1899 nM T62460 C7WO4A 66604791 IC50 = 41 nM T62460 CW53KR 66604810 IC50 = 339 nM T62460 CNW05G 66604855 IC50 = 31 nM T62460 C0JS8O 66604914 IC50 = 5.7 nM T62460 CW9LD1 66604921 IC50 = 62 nM T62460 CTMX20 66605009 IC50 = 31 nM T62460 CP0DB1 66605115 IC50 = 77 nM T62460 CB1WC9 66605298 IC50 = 158 nM T62460 CCWU74 66605322 IC50 = 29 nM T62460 C7Q8ZG 66605359 IC50 = 218 nM T62460 C16TEK 66605475 IC50 = 100 nM T62460 C7MOJ6 66605487 IC50 = 195 nM T62460 CDZA70 66605639 IC50 = 432 nM T62460 C53NBQ 66605756 IC50 = 45 nM T62460 C5PVB2 67008690 IC50 = 2076 nM T62460 C8OZ6W 67008828 IC50 = 863 nM T62460 C1HSE0 67035086 IC50 = 260 nM T62460 CWI6K5 67035106 IC50 > 10000 nM T62460 C38RGB 67035556 IC50 > 10000 nM T62460 CV3HW2 67035568 IC50 > 10000 nM T62460 CZX1E0 67123420 IC50 > 10000 nM T62460 C0RCI2 67123577 IC50 = 5.5 nM T62460 CV63UL 67240318 IC50 > 10000 nM T62460 C78TXA 67277273 IC50 = 110 nM T62460 C0O7TC 67277276 IC50 = 1.5 nM T62460 C3YK7Q 67277763 IC50 = 300 nM T62460 CF4AB0 67277979 IC50 = 2900 nM T62460 C5U2IW 67278045 IC50 = 430 nM T62460 CS9K0L 67278047 IC50 = 140 nM T62460 C2FW8H 67278142 IC50 = 90 nM T62460 CQRS42 67278151 IC50 = 230 nM T62460 C5V9DZ 67278165 IC50 = 520 nM T62460 CMJ29W 67278195 IC50 = 1000 nM T62460 CVL35U 67278385 IC50 = 110 nM T62460 CKVB79 67278425 IC50 = 28 nM T62460 C2C1RE 67329237 IC50 = 41 nM T62460 CV80IQ 67330694 IC50 = 29 nM T62460 CKMV48 67345882 Ki = 0.8 nM T62460 C16THB 67351896 Ki = 12 nM T62460 CXU7P1 67352101 Ki = 16 nM T62460 C4D9NB 67352386 Ki = 8.4 nM T62460 CFX84K 67352945 Ki = 5.9 nM T62460 C1FLT6 67354280 Ki = 120 nM T62460 C9WY2P 67383875 Ki = 24 nM T62460 C14RKJ 67479440 IC50 = 307 nM T62460 C5WQC2 67502257 IC50 > 1000 nM T62460 CX6S4E 68254533 IC50 = 1500 nM T62460 CYMN23 68260892 Ki = 5.4 nM T62460 C4U1IR 68291322 IC50 = 21 nM T62460 C2P7DB 68291391 IC50 = 71 nM T62460 CRM3S0 68291627 IC50 = 100 nM T62460 C4LKB3 68291752 IC50 = 9 nM T62460 CQ49HB 68291755 IC50 = 5 nM T62460 CXI4L1 68291797 IC50 = 41 nM T62460 C8T5VB 68291830 IC50 = 19 nM T62460 CPRW18 68291866 IC50 = 214 nM T62460 C6UWI3 68291981 IC50 = 34 nM T62460 CYN89R 68292156 IC50 = 61 nM T62460 C76EZC 68292170 IC50 = 62 nM T62460 CGA0W6 68292183 IC50 = 15 nM T62460 C93LZT 68292196 IC50 = 190 nM T62460 C8I7GC 68293638 IC50 > 10000 nM T62460 CD56XK 68293660 IC50 > 10000 nM T62460 CYI75G 68678653 IC50 > 30000 nM T62460 C5DGR9 69036886 IC50 = 10000 nM T62460 CK8DC3 69046862 IC50 = 24 nM T62460 COX56A 69809432 IC50 = 189 nM T62460 CECG39 69809726 IC50 = 103 nM T62460 C92EAC 69811936 IC50 = 71 nM T62460 C0XO1M 69812740 IC50 = 113 nM T62460 CASQ98 70650259 IC50 = 1700 nM T62460 CQ2F8J 70824464 Ki = 2600 nM T62460 CJQA59 70929300 IC50 = 67 nM T62460 CNR2Y9 71061323 IC50 = 54 nM T62460 C51JTW 71061588 IC50 = 9.4 nM T62460 CF69WT 71061828 IC50 = 25 nM T62460 COU2C5 71061858 IC50 = 39 nM T62460 CW9OE6 71061878 IC50 = 12 nM T62460 CK9LZ3 71061981 IC50 = 180 nM T62460 CU1T4P 71061987 IC50 = 41 nM T62460 CJH94D 71062030 IC50 = 5.5 nM T62460 CUW46K 71062043 IC50 = 49 nM T62460 C05VNE 71062076 IC50 = 31 nM T62460 C4AC9U 71212257 IC50 < 0.2 nM T62460 CHO4J2 71212467 Ki = 5.4 nM T62460 C7Y2LB 71230234 Ki = 2 nM T62460 CV0U3C 71230392 Ki = 3 nM T62460 COR71Z 71285696 IC50 = 17 nM T62460 C3ZL5S 71285760 IC50 = 64 nM T62460 CME92O 71285933 IC50 = 10 nM T62460 C2FL6H 71286084 IC50 = 5.5 nM T62460 C14YOJ 71286184 IC50 = 12 nM T62460 CX23BP 71288497 IC50 = 22 nM T62460 CH1AJ3 71288512 IC50 = 0.8 nM T62460 CA1T5H 71288539 IC50 = 38 nM T62460 CYU2Z4 71288594 IC50 = 61 nM T62460 CBY4K0 71288602 IC50 = 31 nM T62460 CWLC45 71288607 IC50 = 51 nM T62460 CDST08 71288618 IC50 = 73 nM T62460 C45HTF 71288693 IC50 = 1 nM T62460 COC20B 71288707 IC50 = 370 nM T62460 C6JD3S 71288724 IC50 = 4.6 nM T62460 COV78A 71288729 IC50 = 16 nM T62460 C8DY1N 71288732 IC50 = 61 nM T62460 C6XVG4 71452457 Ki = 24 nM T62460 CY2CE5 71454218 Ki = 5.3 nM T62460 CPO7Y1 71454973 Ki = 2.8 nM T62460 CB8DN6 71455970 Ki = 43 nM T62460 C70KIC 71455971 Ki = 28 nM T62460 CQ0G3P 71455972 Ki = 10 nM T62460 C8LBN3 71457772 Ki = 13 nM T62460 C9HC1M 71457773 Ki = 0.3 nM T62460 C26IQP 71459692 Ki = 2.1 nM T62460 C7GUC2 71461373 Ki = 3.8 nM T62460 CQT1P4 71461404 Ki = 5.8 nM T62460 CTX94J 71461405 Ki = 4.2 nM T62460 CON21P 71463137 Ki = 12 nM T62460 CZPQ54 71463138 Ki = 3.3 nM T62460 CCN01X 71547862 IC50 > 10000 nM T62460 CVEO06 71558636 IC50 = 262 nM T62460 C07SFW 71600166 IC50 = 11600 nM T62460 CWJ1G4 71600167 IC50 = 863 nM T62460 CVYS15 71617859 IC50 = 28 nM T62460 C7T5LI 71655637 Ki = 745 nM T62460 CT3M4B 71655638 Ki = 198 nM T62460 CSC81X 71655639 Ki = 21 nM T62460 CGO74N 71655708 Ki > 3763 nM T62460 C3U1ZV 71655709 Ki = 4.7 nM T62460 CE1JQ3 71655774 Ki = 12 nM T62460 CX5OU4 71681533 Ki = 3.5 nM T62460 C29FVT 71681534 Ki = 10 nM T62460 C7WQP2 71681535 Ki = 13 nM T62460 CEQM71 71681536 Ki = 16 nM T62460 CV5FB0 71681691 Ki = 1.8 nM T62460 C6JH7K 71681692 Ki = 7.2 nM T62460 C30RQG 71681693 Ki = 2.6 nM T62460 C7D8YL 71681694 Ki = 3.4 nM T62460 CE02VF 71681695 Ki = 2 nM T62460 C64WZP 71681852 Ki = 43 nM T62460 C5N6SR 71681853 Ki = 31 nM T62460 CK93ML 71681854 Ki = 1.1 nM T62460 C5E4OF 71682024 Ki = 1.2 nM T62460 C5QK6S 71727668 IC50 = 23 nM T62460 C8PSM2 71737832 Ki = 235 nM T62460 CW52BU 71943288 IC50 = 33000 nM T62460 C54XWG 72190869 IC50 > 10000 nM T62460 C1N7LQ 72202249 IC50 = 5.1 nM T62460 C6THF4 72374600 Ki = 430 nM T62460 CHK46S 72375658 Ki = 98 nM T62460 COPS30 72375659 Ki = 710 nM T62460 CB9ZL4 72375660 Ki = 120 nM T62460 C0K5IO 72375661 Ki = 75 nM T62460 C7PG8Z 72375662 Ki = 398 nM T62460 CCZO42 72375759 Ki = 644 nM T62460 CEV9X5 72375760 Ki = 151 nM T62460 COE6R4 72375761 Ki = 893 nM T62460 C1G8RD 72375763 Ki = 720 nM T62460 C8SLE9 72375764 Ki = 610 nM T62460 C74WLS 72375765 Ki = 3500 nM T62460 CP2KL5 72375766 Ki > 5600 nM T62460 CT9D3J 72375844 Ki = 2800 nM T62460 CZN81X 72375845 Ki = 453 nM T62460 CXL52K 72375846 Ki = 1200 nM T62460 CAV52F 72375847 Ki = 408 nM T62460 C3QT2E 72375850 Ki = 65 nM T62460 C0UJ9M 72375852 Ki = 151 nM T62460 CNJ03L 72375990 Ki > 3500 nM T62460 C5R0WV 72375991 Ki > 3500 nM T62460 CVUL48 72375992 Ki = 2000 nM T62460 CO8KW2 72375993 Ki > 3500 nM T62460 CN0I2W 72375994 Ki > 3500 nM T62460 C1XD7U 72375995 Ki > 3500 nM T62460 C8BJ4U 72375996 Ki > 3500 nM T62460 C7XFW2 72375997 Ki > 3500 nM T62460 CJB95D 72375998 Ki > 3500 nM T62460 CS5V9L 72376089 Ki > 3500 nM T62460 C37GPL 72376090 Ki > 3500 nM T62460 C9U3WO 72376091 Ki > 3500 nM T62460 CK7F6U 72700776 Ki = 3 nM T62460 CLOE10 72706962 IC50 = 1620 nM T62460 CXD38C 73346480 Ki = 2 nM T62460 C0G5RD 73347974 Ki = 661 nM T62460 CRAW59 73349195 Ki = 1100 nM T62460 C41ZJV 73349520 Ki = 4.6 nM T62460 CJE73Y 73352545 Ki = 280 nM T62460 CPRD59 73352546 Ki = 13 nM T62460 CXT70E 73354035 Ki = 380 nM T62460 CGI13D 73354036 Ki = 313 nM T62460 CL4SD8 73355260 Ki > 3500 nM T62460 CMR72H 73355566 Ki = 440 nM T62460 CPT46O 73355567 Ki = 3200 nM T62460 C04CXF 73355568 Ki = 65 nM T62460 C3G2BM 73357112 Ki = 18 nM T62460 CO6F2B 73357113 Ki = 7 nM T62460 CS41CX 75108409 IC50 = 131 nM T62460 CO0BQ5 76310565 IC50 = 628 nM T62460 C6ZAB2 76310566 IC50 > 10000 nM T62460 C0F6VU 76310567 IC50 = 300 nM T62460 CDO38G 76310568 IC50 > 10000 nM T62460 CL42BQ 76310569 IC50 > 10000 nM T62460 CWI1Q4 76310570 IC50 = 564 nM T62460 C8OY6Q 76310785 IC50 > 100000 nM T62460 CAL3U7 76310788 IC50 > 100000 nM T62460 C7SXJ1 76314208 IC50 = 1060 nM T62460 CSDI71 76314209 IC50 > 10000 nM T62460 C12YAE 76314414 IC50 > 100000 nM T62460 CXF1I3 76317774 IC50 = 4903 nM T62460 CY79VS 76317775 IC50 > 10000 nM T62460 CNK2I1 76317776 IC50 > 10000 nM T62460 CS02NA 76317777 IC50 = 1784 nM T62460 CAHW32 76317778 IC50 = 4819 nM T62460 C97RBS 76317979 IC50 > 100000 nM T62460 C2SMK1 76321491 IC50 > 10000 nM T62460 C2DSX7 76321492 IC50 = 4097 nM T62460 CXA4O1 76325093 IC50 > 10000 nM T62460 CEZ64F 76325209 IC50 = 22 nM T62460 C1AI0J 76325315 IC50 > 100000 nM T62460 CPQA45 76325323 IC50 > 100000 nM T62460 C8GK0H 76328659 IC50 = 11120 nM T62460 CJN89E 76332335 IC50 > 10000 nM T62460 CW1QK4 76332336 IC50 = 423 nM T62460 C2P1MX 76332338 IC50 = 2174 nM T62460 CB5Y0Z 76332540 IC50 > 100000 nM T62460 CB4KQ7 76335967 IC50 = 8640 nM T62460 C84PFQ 76335968 IC50 = 2058 nM T62460 CW1HQ9 76370451 IC50 = 3.9 nM T62460 CD6Y1F 78320046 IC50 = 40 nM T62460 CW08SU 78320048 IC50 = 9 nM T62460 CWI93D 78323836 IC50 = 22 nM T62460 C5UK9L 78323837 IC50 = 14 nM T62460 CQ3EJ1 78324132 IC50 = 28 nM T62460 C7VOX0 78324136 IC50 = 42 nM T62460 CA2Y8L 78324435 IC50 = 51 nM T62460 C4I7WD 78324744 IC50 = 22 nM T62460 CQ2SU8 78673832 IC50 > 30000 nM T62460 CE0W9R 78673833 IC50 > 30000 nM T62460 CPG3A5 86302574 IC50 > 30000 nM T62460 C96EDF 86660048 IC50 = 1000 nM T62460 CC8I0M 86707711 IC50 = 1.9 nM T62460 CW4Z2F 89470642 IC50 = 0.15 nM T62460 CBRF87 89470690 IC50 = 0.24 nM T62460 C7B8OH 89470730 IC50 = 14 nM T62460 CHUO79 89471082 IC50 = 3 nM T62460 CDQ8C6 89471114 IC50 = 0.13 nM T62460 C4G5LP 89471136 IC50 = 33 nM T62460 CX1DZ3 89471497 IC50 = 0.3 nM T62460 CX1MA3 89471556 IC50 = 1.2 nM T62460 C1HW4B 89735655 IC50 = 4300 nM T62460 CG9C6J 89765129 IC50 = 48 nM T62460 C13GOX 89775209 IC50 = 90 nM T62460 C3N6RU 89775221 IC50 = 30 nM T62460 CG5P9A 90153688 IC50 > 50000 nM T62460 CTV52A 90367281 IC50 = 1.5 nM T62460 CY0UC4 90645194 IC50 > 10000 nM T62460 C7EXH8 91755097 IC50 = 0.7 nM T62460 C37IZB 91755098 IC50 = 1.3 nM T62460 C7UAK5 91809175 IC50 > 2000 nM T62460 C8RG6H 91827514 IC50 = 1900 nM T62460 C0Y8ZK 91933875 IC50 > 1000 nM T62460 C64SIO 92042864 IC50 = 896 nM T62460 C9BL4M 92045136 IC50 = 22 nM T62460 CXU1Z2 101043725 IC50 > 2000 nM T62460 C9G5TC 102515538 Ki = 172 nM T62460 CM2C3W 105539869 IC50 = 130 nM T62460 C3ECY5 117625437 IC50 = 16 nM T62460 CZC84D 117769161 IC50 = 1.2 nM T62460 CE7BZ8 117769174 IC50 = 28 nM T62460 CBJ07Q 117769217 IC50 = 3.6 nM T62460 CXHQ08 117769229 IC50 = 1 nM T62460 CS9WO4 117769234 IC50 = 0.9 nM T62460 C61VXQ 117769241 IC50 = 0.9 nM T62460 C1SA9I 117769244 IC50 = 2.2 nM T62460 C0VY7C 117769271 IC50 = 0.5 nM T62460 C6O9BT 117769272 IC50 = 7.2 nM T62460 CSR9B0 117769289 IC50 = 1.2 nM T62460 C2M9CR 117769307 IC50 = 3.3 nM T62460 C7FWS3 117769309 IC50 = 0.9 nM T62460 CYWV32 117769339 IC50 = 6.6 nM T62460 CZV35K 117769346 IC50 = 1.7 nM T62460 C5V6RG 117769349 IC50 = 4.9 nM T62460 C4O1PX 117769362 IC50 = 1.2 nM T62460 CPV4C8 117769365 IC50 = 0.6 nM T62460 CP3MC5 117769379 IC50 = 1.2 nM T62460 C8V6LG 117769392 IC50 = 2 nM T62460 C2NBZ8 117769396 IC50 = 1.3 nM T62460 COV59Y 117769408 IC50 = 0.7 nM T62460 CXJ3I6 117769409 IC50 = 4 nM T62460 C8LTZ6 117769464 IC50 = 2.4 nM T62460 C4KL1Y 117769470 IC50 = 0.8 nM T62460 CQ46WT 117769476 IC50 = 2.3 nM T62460 CSKO30 117769533 IC50 = 6.6 nM T62460 C6XC3W 117769575 IC50 = 0.4 nM T62460 CS95HO 117769592 IC50 = 0.8 nM T62460 C0PIL5 117769623 IC50 = 1.6 nM T62460 CO3DA2 117769866 IC50 = 6.9 nM T62460 CI46CP 117770056 IC50 = 230 nM T62460 C7NI8L 117770083 IC50 = 100 nM T62460 CJ3QC8 117770200 IC50 = 3100 nM T62460 CSD47C 117770482 IC50 = 15 nM T62460 C8SNB9 117770595 IC50 = 91 nM T62460 CJ1V9A 117770654 IC50 = 65 nM T62460 CS8E6M 117770678 IC50 = 370 nM T62460 CM7X9N 117770754 IC50 = 79 nM T62460 C4CFG6 117770831 IC50 = 260 nM T62460 C0X1EQ 117809257 IC50 = 26 nM T62460 CDUH09 117809287 IC50 = 0.6 nM T62460 C8HYU9 117926195 IC50 > 10000 nM T62460 CGQK96 118115537 IC50 = 984 nM T62460 C2OX1Q 118115706 IC50 = 274 nM T62460 CWCO47 118115913 IC50 = 2290 nM T62460 C72LYV 118116131 IC50 = 1400 nM T62460 C4JW5D 118116385 IC50 = 1150 nM T62460 CNX7M9 118473558 IC50 > 2000 nM T62460 CK6Z8O 118475621 IC50 = 49 nM T62460 CIVS69 118475644 IC50 = 11 nM T62460 C17FYA 118475649 IC50 = 495 nM T62460 CE49ZI 118475652 IC50 = 35 nM T62460 C65NIK 118475658 IC50 = 656 nM T62460 C0A9RJ 118475705 IC50 = 24.4 nM T62460 CWQ36P 118475893 IC50 = 731 nM T62460 CN04RH 118475894 IC50 > 3000 nM T62460 C2P0CG 118475938 IC50 = 743 nM T62460 CJYV54 118494221 IC50 > 1000 nM T62460 CLTV08 118690376 IC50 = 16 nM T62460 CRK6J2 118690573 IC50 = 67 nM T62460 CTR74C 118690690 IC50 = 24 nM T62460 CY7BI2 118706214 IC50 > 10000 nM T62460 C2C0AG 118707521 IC50 > 100000 nM T62460 C2DJA0 118707522 IC50 > 100000 nM T62460 CBF28W 118707523 IC50 > 100000 nM T62460 CQ6ON4 118707525 IC50 > 100000 nM T62460 C38UWP 118707526 IC50 > 100000 nM T62460 C64ZQX 118707543 IC50 > 100000 nM T62460 CX58DI 118716791 IC50 > 30000 nM T62460 CD9X2B 118716796 IC50 > 30000 nM T62460 C2YJ0O 118716797 IC50 > 30000 nM T62460 CL3UO9 118716798 IC50 > 30000 nM T62460 C71BAM 118716799 IC50 > 30000 nM T62460 CU4EL6 118716806 IC50 > 30000 nM T62460 CP0IO9 118722564 IC50 = 2225 nM T62460 C5K2QD 118723914 IC50 = 48 nM T62460 C59YJC 118723915 IC50 = 24 nM T62460 C2ON7Y 118723916 IC50 = 270 nM T62460 C5U8WG 118723917 IC50 = 56 nM T62460 C0ZMR8 118723918 IC50 = 67 nM T62460 C4Z5LJ 118723919 IC50 = 150 nM T62460 C85ELI 118723920 IC50 = 50 nM T62460 CGW49X 118723921 IC50 = 110 nM T62460 CXC8K9 118723922 IC50 = 270 nM T62460 CR5JD8 118723923 IC50 = 84 nM T62460 C9W1BU 118723924 IC50 = 250 nM T62460 C2K0MN 118724183 IC50 > 10000 nM T62460 C0G8DY 118724184 IC50 > 10000 nM T62460 CYN2Q5 118724185 IC50 > 10000 nM T62460 C5LR9P 118724186 IC50 = 5740 nM T62460 CXUE02 118724187 IC50 > 10000 nM T62460 C2IYQ8 118724188 IC50 = 413 nM T62460 CQEM50 118724189 IC50 > 10000 nM T62460 C38URV 118724190 IC50 = 371 nM T62460 CDI46A 118724191 IC50 = 2554 nM T62460 C9MG2U 118724192 IC50 = 572 nM T62460 CDH50E 118724193 IC50 > 10000 nM T62460 C7AE5B 118724194 IC50 = 3012 nM T62460 CS61RK 118724197 IC50 = 3098 nM T62460 C6LTE8 118724198 IC50 = 0.6 nM T62460 CP1HW5 118724199 IC50 = 8.3 nM T62460 CR8P2W 118724200 IC50 = 147 nM T62460 CW2G9E 118724201 IC50 = 16 nM T62460 C8JGN7 118868847 IC50 = 19 nM T62460 C3DK1Q 118868914 IC50 = 10 nM T62460 CQ1TL7 118879520 IC50 = 90 nM T62460 CAZO34 118911466 IC50 = 470 nM T62460 C6VAE4 118911477 IC50 = 9 nM T62460 CRQV39 118911480 IC50 = 20 nM T62460 C5Z0XH 118911481 IC50 = 8.5 nM T62460 CG0T1W 118911482 IC50 = 170 nM T62460 COD91F 118911483 IC50 = 230 nM T62460 C5LYI2 118911484 IC50 = 160 nM T62460 CA9P3K 118911491 IC50 = 31 nM T62460 CB81YO 118911492 IC50 = 12 nM T62460 C2DG5M 118911497 IC50 = 1400 nM T62460 CI2EU5 118911501 IC50 = 100 nM T62460 CA3EF6 118911506 IC50 = 20 nM T62460 C9BE2G 118911507 IC50 = 520 nM T62460 C75DOY 118911508 IC50 = 16 nM T62460 CZ3D0U 118911512 IC50 = 420 nM T62460 C1AE4J 118911514 IC50 = 40 nM T62460 CN53SL 118911517 IC50 = 21 nM T62460 CCX4J8 118911542 IC50 = 74 nM T62460 C7R0NJ 118911545 IC50 = 120 nM T62460 CIS3Z5 118911549 IC50 = 1.4 nM T62460 C49PME 118911551 IC50 = 1500 nM T62460 CJT3P9 118911552 IC50 = 120 nM T62460 CX01BU 118911553 IC50 = 170 nM T62460 C0TU7V 118911556 IC50 = 26 nM T62460 C0TX7B 118911557 IC50 = 23 nM T62460 CYI3O6 118911558 IC50 = 15 nM T62460 C28MLV 118911560 IC50 = 53 nM T62460 C49UGI 118911561 IC50 = 34 nM T62460 C9LD1H 118911562 IC50 = 190 nM T62460 CTR8D0 118911563 IC50 = 77 nM T62460 CY5EN8 118911565 IC50 = 6.3 nM T62460 C84BPW 118911566 IC50 = 6.9 nM T62460 CT4MJ8 118911570 IC50 = 5.8 nM T62460 C2AZP5 118911571 IC50 = 9.8 nM T62460 CQ59WD 118911572 IC50 = 29 nM T62460 C2S7MO 118911575 IC50 = 9.4 nM T62460 C45HFX 118911579 IC50 = 500 nM T62460 CCSH64 118911580 IC50 = 150 nM T62460 CB48OQ 118911581 IC50 = 12 nM T62460 CZY2V6 118911582 IC50 = 670 nM T62460 C2PA8M 118911583 IC50 = 13 nM T62460 C70XKA 118911584 IC50 = 180 nM T62460 CD9C1A 118911585 IC50 = 75 nM T62460 CRZ20W 118911587 IC50 = 7.2 nM T62460 CTQ4J9 118911588 IC50 = 9.3 nM T62460 C3QKH8 118911601 IC50 = 17 nM T62460 COY26N 118911635 IC50 = 140 nM T62460 CL3C9A 118911638 IC50 = 69 nM T62460 CN4O2C 118911639 IC50 = 50 nM T62460 C9O4WL 118911640 IC50 = 54 nM T62460 C3SE0K 118911642 IC50 = 85 nM T62460 C5LHC4 118911643 IC50 = 2.8 nM T62460 CPK30A 118911645 IC50 = 790 nM T62460 CYTV80 121284861 IC50 > 2000 nM T62460 CY9M5S 122182022 IC50 = 29 nM T62460 C2MCH6 122182157 IC50 = 84 nM T62460 CK4A6L 122182159 IC50 = 11 nM T62460 CFU15S 122191618 IC50 = 65 nM T62460 CE4F3A 122191619 IC50 = 1700 nM T62460 CAC5U1 122191620 IC50 = 220 nM T62460 CRF2K0 122191625 IC50 = 540 nM T62460 CPY1K9 122191778 IC50 = 2728 nM T62460 C1H4IX 122192065 IC50 = 6100 nM T62460 C98EJO 122192066 IC50 = 11300 nM T62460 CM1XD7 122192067 IC50 = 100 nM T62460 C0MLH5 122192068 IC50 = 2200 nM T62460 CC4T6A 122192069 IC50 = 5700 nM T62460 CGO6M7 122192070 IC50 = 4300 nM T62460 CBP34K 122192071 IC50 = 11600 nM T62460 CA2TF6 122192072 IC50 = 18200 nM T62460 CFY30Z 122192073 IC50 = 2900 nM T62460 CJ09XF 122192074 IC50 = 3700 nM T62460 C6LS8X 122192075 IC50 = 3100 nM T62460 C7DJA5 122192076 IC50 = 9300 nM T62460 CAS86F 122192079 IC50 = 32400 nM T62460 CG7TP0 122192080 IC50 = 8100 nM T62460 C5K8UM 122192081 IC50 = 3400 nM T62460 CS4XB9 122199230 IC50 = 90 nM T62460 CNA45R 122362931 IC50 = 19 nM T62460 CW9BU8 126643886 IC50 = 29 nM T62460 C4BJ8G 126645320 IC50 = 10 nM T62460 CL60VJ 126647240 IC50 = 270 nM T62460 C1XS8H 126647348 IC50 = 3.6 nM T62460 CSJ1G7 126647349 IC50 = 650 nM T62460 C9QCD3 126715362 IC50 < 4 nM T62460 CNPB25 126715363 IC50 = 7600 nM T62460 CY7US6 126715366 IC50 = 120 nM T62460 CJS53A 126715367 IC50 < 6 nM T62460 CX37RN 126715380 IC50 = 70 nM T62460 C2DQU9 126715387 IC50 = 643 nM T62460 CH6YP0 126715392 IC50 = 130 nM T62460 C1QB5R 126715400 IC50 = 7 nM T62460 CG7YQ2 126715454 IC50 < 3 nM T62460 CO2X6J 126715460 IC50 = 8 nM T62460 CR9C1G 127030133 IC50 = 22 nM T62460 CU4AJ8 127037981 IC50 = 317 nM T62460 CA0O1B 127037982 IC50 = 274 nM T62460 C50NKB 127037983 IC50 = 12200 nM T62460 CF8KQ6 127038326 IC50 = 832 nM T62460 C5WV8P 127038327 IC50 = 356 nM T62460 CI8ZB6 127038328 IC50 = 4910 nM T62460 C98DQZ 127038947 IC50 = 173 nM T62460 CQ4OE5 127039917 IC50 = 801 nM T62460 CC1XP0 127040339 IC50 = 199 nM T62460 C8H7JN 127040340 IC50 = 177 nM T62460 CRQS46 127040341 IC50 > 30000 nM T62460 C3B0AP 127040342 IC50 = 4510 nM T62460 C7KLD9 127040660 IC50 = 977 nM T62460 C4JF8H 127040661 IC50 = 4.9 nM T62460 CC9J7R 127040662 IC50 = 34 nM T62460 CP1RY4 127040993 IC50 = 9 nM T62460 C7P5MY 127040994 IC50 = 49 nM T62460 CB23SC 127041238 IC50 = 561 nM T62460 CJ7QW5 127041248 IC50 = 73 nM T62460 C1N6BC 127041249 IC50 = 36 nM T62460 C5SLH0 127041250 IC50 = 275 nM T62460 C28YFA 127041251 IC50 > 30000 nM T62460 CIP84Z 127041549 IC50 = 5230 nM T62460 CQP76E 127041550 IC50 = 2100 nM T62460 C3A1VL 127041551 IC50 > 30000 nM T62460 CEJ97D 127041858 IC50 = 17 nM T62460 C35OPG 127041859 IC50 = 177 nM T62460 CEN15W 127041860 IC50 = 138 nM T62460 C4UBE5 127041861 IC50 = 872 nM T62460 C7Q5YC 127045965 IC50 = 670 nM T62460 CB2SE8 127049004 IC50 = 5300 nM T62460 CS6ZO5 127049005 IC50 = 5400 nM T62460 C1PE9L 127050562 IC50 = 80 nM T62460 CZ5D8C 127050563 IC50 = 7000 nM T62460 CX46RS 127050564 IC50 = 2000 nM T62460 C3LI1J 127050565 IC50 = 150 nM T62460 CG91WC 127052080 IC50 = 90 nM T62460 C0FM1R 130196825 IC50 = 787 nM T62460 CZ13WL 130339268 IC50 = 383 nM T62460 CD4NY1 131839645 IC50 = 0.1 nM T62460 CUO0C5 132156633 IC50 > 10000 nM T62460 CK4FI7 132277003 IC50 = 966 nM T62460 C5CZA1 132578411 IC50 = 444 nM T62460 C75NKQ 134537028 IC50 = 26 nM T62460 CPDT50 134537033 IC50 = 110 nM T62460 C8CKE5 134537037 IC50 = 510 nM T62460 C7H8QW 134537039 IC50 = 19 nM T62460 C0ZY5J 134537043 IC50 = 25 nM T62460 CJDM08 134537050 IC50 = 66 nM T62460 CQ7G4C 134537056 IC50 = 4.1 nM T62460 CQ1NX6 134537061 IC50 = 740 nM T62460 C43CFZ 134537067 IC50 = 170 nM T62460 CELH87 134537071 IC50 = 34 nM T62460 C8DAO7 134537074 IC50 = 1.9 nM T62460 CQ9OU1 134537081 IC50 = 140 nM T62460 CH78PN 134537085 IC50 = 160 nM T62460 CN5P0G 134537092 IC50 = 260 nM T62460 CHY1S4 134537094 IC50 = 110 nM T62460 C8L7UN 134537111 IC50 = 11 nM T62460 C42TFN 134537113 IC50 = 13 nM T62460 C58HUF 134537114 IC50 = 53 nM T62460 C3LRB2 134537119 IC50 = 22 nM T62460 CWU3Z2 134537141 IC50 = 52 nM T62460 CEOW01 134537147 IC50 = 17 nM T62460 C0T7VN 134537152 IC50 = 79 nM T62460 CZD72H 134537156 IC50 = 11 nM T62460 C3HC0S 134537158 IC50 = 11 nM T62460 CTP15L 134537160 IC50 = 70 nM T62460 C6Z9QY 134537161 IC50 = 28 nM T62460 C9ME6L 134537163 IC50 = 14 nM T62460 CEQ15Z 134537167 IC50 = 70 nM T62460 C8N6ZF 134537169 IC50 = 9.5 nM T62460 CXA39D 134537177 IC50 = 19 nM T62460 C97OTS 134537185 IC50 = 62 nM T62460 CHK0V4 134611545 IC50 = 0.14 nM T62460 C20FAE 134611548 IC50 = 0.37 nM T62460 C51PKU 134611580 IC50 = 0.22 nM T62460 CN75GU 134611727 IC50 = 12 nM T62460 C80PJI 134611728 IC50 = 16 nM T62460 C2AN7T 134611886 IC50 > 100000 nM T62460 CFM46L 134812674 IC50 = 358 nM T62460 C2VC5Y 134817793 IC50 < 3 nM T62460 CVF86X 135125189 IC50 = 0.07 nM T62460 C9MCQ0 135138184 IC50 = 0.4 nM T62460 C7V2MJ 135142423 IC50 = 0.54 nM T62460 CLET52 135142442 IC50 = 0.3 nM T62460 CU13RW 135142625 IC50 = 1.2 nM T62460 CM7N0J 135142656 IC50 = 0.92 nM T62460 CG6JI9 135142885 IC50 = 0.25 nM T62460 CQD32R 135143120 IC50 = 0.49 nM T62460 C7PJ6X 135566704 IC50 > 30000 nM T62460 CPHG43 135567142 IC50 = 0.1 nM T62460 C2NRS8 135567293 IC50 = 0.4 nM T62460 C4R1FH 135567294 IC50 = 1.7 nM T62460 CA0R9G 135567295 IC50 = 60 nM T62460 CRI5F3 135839295 IC50 = 6.1 nM T62460 CH8W7B 135839328 IC50 = 68.6 nM T62460 CD32NI 135894059 IC50 = 1351 nM T62460 CJID74 136013449 EC50 = 350 nM T62460 CHA4N2 136013680 IC50 > 10 nM T62460 C1DNM8 136048702 IC50 = 0.7 nM T62460 CL53YD 136048703 IC50 = 0.5 nM T62460 C8PFY0 136048704 IC50 = 0.3 nM T62460 CKC87M 136048705 IC50 = 3.2 nM T62460 C8TA5Y 136048706 IC50 = 26 nM T62460 CM2A3P 136048707 IC50 = 1.6 nM T62460 C76OBL 136048708 IC50 = 5 nM T62460 C75UYC 136048709 IC50 = 5 nM T62460 CA10UT 136048710 IC50 = 10 nM T62460 C1YUD0 136219394 IC50 > 10 nM T62460 CIU8W3 136254389 IC50 > 10 nM T62460 C1P6ZW 136263939 IC50 < 0.1 nM T62460 C0R2IL 136901416 IC50 = 4.365 nM T62460 C5JIR2 136987005 IC50 > 100000 nM T62460 CIJ71W 137028350 IC50 = 100 nM T62460 CS15TL 137028351 IC50 = 3100 nM T62460 CH3M4B 137083628 IC50 > 30000 nM T62460 CJA07O 137083629 IC50 > 30000 nM T62460 C9F8PX 137083630 IC50 > 30000 nM T62460 CE9V4U 137174991 IC50 = 2 nM T62460 C2FLS4 137175037 IC50 = 2 nM T62460 C6V7OD 137175063 IC50 = 0.8 nM T62460 C2KF1R 137175070 IC50 = 3 nM T62460 C5XJ4Q 137175071 IC50 = 6 nM T62460 CA3E0R 137175072 IC50 = 13 nM T62460 C4WET8 137175109 IC50 = 0.4 nM T62460 CM64UH 137175110 IC50 = 0.8 nM T62460 CQX1H3 137175111 IC50 = 1.3 nM T62460 C0YBL9 137175112 IC50 = 7 nM T62460 CP7RH5 137175113 IC50 = 8 nM T62460 CJ94DH 137175128 IC50 = 0.9 nM T62460 C70DIP 137223928 IC50 = 1.8 nM T62460 C9F3KV 137321155 IC50 = 3.37 nM T62460 CJK67W 137321156 IC50 = 125.1 nM T62460 C3Z4AT 137321159 IC50 = 2703 nM T62460 CMY0V2 137321160 IC50 = 422 nM T62460 CWM9S4 137349398 IC50 = 5 nM T62460 CAM8K0 137632226 IC50 = 85 nM T62460 CH9WK1 137632228 IC50 = 1100 nM T62460 C7R2HI 137632648 IC50 = 11 nM T62460 C2I3PY 137633211 IC50 = 264 nM T62460 CJN68H 137633647 IC50 = 10 nM T62460 CF6RH5 137633780 IC50 = 0.04 nM T62460 COE76K 137634328 IC50 = 2.1 nM T62460 C6IU0M 137634461 IC50 = 0.9 nM T62460 CE4DH3 137635161 IC50 = 31 nM T62460 C6JVG9 137635398 IC50 = 17 nM T62460 CMV38W 137635509 IC50 = 1422 nM T62460 CM73AT 137635759 IC50 = 17 nM T62460 CH5SI7 137636771 IC50 = 19 nM T62460 C8I2NQ 137637573 IC50 = 196 nM T62460 C3RF7B 137638414 IC50 = 141 nM T62460 CE0ZF8 137638897 IC50 = 1.3 nM T62460 C50WHR 137641404 IC50 = 39 nM T62460 C2VWE5 137642024 IC50 = 37 nM T62460 CJ6PU9 137642141 IC50 = 2.3 nM T62460 C0RX1Z 137642404 IC50 = 0.4 nM T62460 C9GDQ6 137642740 IC50 = 0.19 nM T62460 C94ELU 137643208 IC50 > 2000 nM T62460 CO83EQ 137643608 IC50 = 26.8 nM T62460 CQP79B 137643915 IC50 = 12 nM T62460 CGHP09 137645020 IC50 = 0.9 nM T62460 CN34SE 137646319 IC50 > 2000 nM T62460 CI8S5A 137646690 IC50 = 144 nM T62460 CGE91V 137646834 IC50 = 36 nM T62460 CE8SH2 137647292 IC50 = 974 nM T62460 CW6D9H 137648009 IC50 = 92 nM T62460 C9KW2L 137648948 IC50 = 123 nM T62460 CHN7A3 137648975 IC50 = 8 nM T62460 CIB60Q 137649981 IC50 = 0.24 nM T62460 CF4X3E 137650150 IC50 = 2756.5 nM T62460 CVHT54 137650515 IC50 = 14 nM T62460 CJQ72A 137650866 IC50 = 863 nM T62460 CA9K6R 137650880 IC50 = 52 nM T62460 COCF21 137651256 IC50 = 6 nM T62460 C3Z7LM 137651481 IC50 = 0.5 nM T62460 CQ27PY 137651710 IC50 = 7.5 nM T62460 CYA52Z 137652173 IC50 = 24 nM T62460 C28QUP 137652864 IC50 > 10000 nM T62460 C6UEB9 137653042 IC50 = 30 nM T62460 CK81UT 137654424 IC50 = 1700 nM T62460 CW6SO7 137654686 IC50 = 178 nM T62460 CCR5B3 137654793 IC50 = 11 nM T62460 CKM89A 137654900 IC50 = 0.18 nM T62460 C26ONG 137654955 IC50 = 5 nM T62460 CP5S6L 137655441 IC50 = 0.6 nM T62460 CVBS03 137656215 IC50 = 0.06 nM T62460 CYWE21 137656346 IC50 = 0.5 nM T62460 C6V3WR 137656619 IC50 = 3 nM T62460 CT1EP3 137656679 IC50 = 9.7 nM T62460 C8VC9A 137657080 IC50 = 0.8 nM T62460 C49GYQ 137658008 IC50 = 21 nM T62460 C59BVH 137658028 IC50 = 0.3 nM T62460 CO6C8I 137658504 IC50 = 11 nM T62460 CW4CK8 137659037 IC50 = 1.4 nM T62460 C86KOS 137659382 IC50 = 6 nM T62460 CR41KW 137660124 IC50 = 0.1 nM T62460 CQ8KF2 137660642 IC50 = 70 nM T62460 COMQ54 137661391 IC50 = 15 nM T62460 CJ52WM 137661888 IC50 = 57 nM T62460 CU2L5H 138108525 IC50 = 52 nM T62460 C2W0JU 138319690 EC50 = 30 nM T62460 C28PJZ 138376574 IC50 = 180 nM T62460 CXV84M 138377596 IC50 = 4.8 nM T62460 C8X9DR 138584993 IC50 = 30.17 nM T62460 C9NL1M 138585023 IC50 = 6.59 nM T62460 CHX6N7 138585027 IC50 = 1.2 nM T62460 C3RM2Z 138585033 IC50 = 4.23 nM T62460 CBF8S4 138585069 IC50 = 616.3 nM T62460 C4O0GC 138585070 IC50 = 9.89 nM T62460 C7KYU3 138585074 IC50 = 43.78 nM T62460 CE5S4Z 138585101 IC50 = 3334 nM T62460 CM63FA 138585111 IC50 = 11.48 nM T62460 C2U8PZ 138585129 IC50 = 1.91 nM T62460 C0Y2WZ 138585150 IC50 = 95.62 nM T62460 CHMX08 138585151 IC50 = 17.86 nM T62460 CA8N5T 138585156 IC50 = 37.54 nM T62460 CG8TR3 138585164 IC50 = 5.28 nM T62460 C3JR7K 138585184 IC50 = 138.1 nM T62460 CQI78V 138585192 IC50 = 10.61 nM T62460 C2UCN9 138605457 IC50 = 103.15 nM T62460 C3RM1U 138605458 IC50 = 423.8 nM T62460 CD4M3W 138605461 IC50 = 58.26 nM T62460 C4VMQ9 138605557 IC50 = 304.45 nM T62460 CQ6R7X 138911330 IC50 > 40000 nM T62460 CI1D9F 139600335 IC50 = 26 nM T62460 CI7C4P 140943115 IC50 > 2000 nM T62460 C7U3KH 140943149 IC50 > 2000 nM T62460 C18QDP 141523774 IC50 = 589.1 nM T62460 CD9F4Y 141523776 IC50 = 168.3 nM T62460 C4L6JD 141523781 IC50 = 361.2 nM T62460 CSZQ36 141523784 IC50 = 140 nM T62460 CTYQ49 141523785 IC50 = 190.4 nM T62460 CU51PI 141531440 IC50 = 694 nM T62460 C81RPA 141531442 IC50 = 1946.9 nM T62460 CAT46B 141531443 IC50 = 618.1 nM T62460 CS37YV 141531444 IC50 = 1372.5 nM T62460 CN75MA 141728817 IC50 = 10 nM T62460 C7EL5X 141728840 IC50 = 14 nM T62460 C9H8PX 141728841 IC50 = 15 nM T62460 CC03XH 141728860 IC50 = 30 nM T62460 CECS13 141753441 IC50 = 1286 nM T62460 C1JR5B 142379949 IC50 = 0.14 nM T62460 C45HDA 142744326 IC50 = 82 nM T62460 CFY17M 142744351 IC50 = 138 nM T62460 CM0BL5 142744356 IC50 = 186 nM T62460 C47YDW 142744361 IC50 = 72 nM T62460 C2L1ZB 142744367 IC50 = 142 nM T62460 CZ6FC4 145362469 IC50 = 16 nM T62460 C2OA9H 145949725 IC50 < 3 nM T62460 CY04PB 145950223 EC50 = 37 nM T62460 CDTW63 145950378 IC50 < 3 nM T62460 CDJ81U 145952312 EC50 = 325 nM T62460 C2XP8N 145953005 IC50 = 29 nM T62460 CN0V3D 145953512 EC50 = 68 nM T62460 C1OQ3J 145953599 IC50 < 3 nM T62460 CNS52L 145954024 EC50 = 189 nM T62460 CRU9F8 145955362 IC50 <= 3 nM T62460 CIP2J9 145955397 IC50 = 55 nM T62460 CQ68WS 145956107 IC50 = 4 nM T62460 CZ0B7A 145956262 IC50 = 13 nM T62460 CO6SV3 145957001 IC50 = 42 nM T62460 C51ADW 145958260 IC50 = 10 nM T62460 C3L8IE 145958641 IC50 = 69 nM T62460 C7B2LD 145959014 IC50 < 3 nM T62460 CO05IK 145959360 IC50 = 76 nM T62460 CMCG17 145959462 IC50 < 3 nM T62460 C2LD5V 145960573 EC50 = 101 nM T62460 CFY21D 145961655 EC50 = 7660 nM T62460 CI9Z7U 145962747 IC50 = 45 nM T62460 CQ86LZ 145963345 IC50 = 117 nM T62460 CEDZ18 145971190 EC50 = 26 nM T62460 CKPM09 145971514 IC50 = 6 nM T62460 C7K1AJ 145971681 IC50 = 359 nM T62460 C7OD0E 145973587 EC50 = 50 nM T62460 CHVD06 145979212 IC50 > 10000 nM T62460 C7L1IC 145979240 IC50 = 4027 nM T62460 CAJ37B 145979552 IC50 = 94 nM T62460 CE31VG 145979714 IC50 = 82 nM T62460 C7N8DU 145980127 IC50 = 814 nM T62460 C8AMK1 145980722 IC50 = 100 nM T62460 C81XFH 145980840 IC50 = 105 nM T62460 C85XBC 145981348 IC50 = 81 nM T62460 C5VF8P 145983087 IC50 = 1067 nM T62460 CS1GK8 145983460 IC50 = 146.8 nM T62460 CG97VS 145983548 IC50 = 496.8 nM T62460 CA20KM 145983867 IC50 = 1354.7 nM T62460 C7THN1 145984160 IC50 = 844 nM T62460 C30EHD 145984172 IC50 = 1720 nM T62460 CP8J3H 145984569 IC50 = 112.3 nM T62460 C42SJR 145984669 IC50 = 496.8 nM T62460 CLH7K9 145984673 IC50 = 165.4 nM T62460 C67HUC 145984822 IC50 = 342.4 nM T62460 CG4U3I 145985120 IC50 = 1674.7 nM T62460 CY7X5L 145986106 IC50 = 2291.5 nM T62460 C03PYD 145986466 IC50 < 1000 nM T62460 C2JCA0 145987101 IC50 = 203 nM T62460 CW7V1O 145987719 IC50 > 50000 nM T62460 C8NEY2 145987871 IC50 = 97 nM T62460 C9ZC0H 145987988 IC50 > 2000 nM T62460 C9KJ1A 145988137 IC50 = 94 nM T62460 C9BX4U 145988956 IC50 = 733 nM T62460 CIVK73 145989244 IC50 = 775 nM T62460 CC8GZ3 145989610 IC50 = 113 nM T62460 C5I8SR 145989639 IC50 = 6501 nM T62460 CIU9W4 145990027 IC50 = 369 nM T62460 C3DWZ0 145990496 IC50 > 4163 nM T62460 CTX1A3 145990814 IC50 = 37 nM T62460 CNG35K 145991262 IC50 = 493 nM T62460 C0M6LD 145991292 IC50 = 1715 nM T62460 CKGE38 145991618 IC50 = 1179 nM T62460 CI8R6P 145992803 IC50 = 1942 nM T62460 CD09RT 145992905 IC50 = 52.1 nM T62460 CG21JZ 145993080 IC50 > 2000 nM T62460 CR2F1Y 145993348 IC50 = 92 nM T62460 C51DMH 145993445 IC50 = 652 nM T62460 C1S2ER 146025986 IC50 = 18 nM T62460 CHQU21 146185142 IC50 = 1223 nM T62460 C71KXB 146185156 IC50 = 82 nM T62460 C9IA1X 146185163 IC50 = 1796 nM T62460 CS0OL6 146185170 IC50 = 660 nM T62460 C1IAH7 146185174 IC50 = 120 nM T62460 C5T7UA 154701267 IC50 = 26 nM T62460 C7PLT9 155510967 IC50 = 7179 nM T62460 C1WRE2 155511764 IC50 = 76 nM T62460 CR1SE8 155511850 IC50 = 3062 nM T62460 C2MD1Q 155513187 IC50 > 10000 nM T62460 CM95KR 155513637 IC50 = 627.1 nM T62460 C83ZSG 155514311 IC50 = 30 nM T62460 C7MJY5 155514805 IC50 = 21 nM T62460 CUIO35 155516044 IC50 = 215 nM T62460 CTP29J 155516678 IC50 = 20 nM T62460 C9VK3I 155517004 IC50 > 2000 nM T62460 C2X8HA 155517088 IC50 > 2000 nM T62460 CE2Q3D 155517448 IC50 = 70 nM T62460 C0E7WS 155518120 IC50 = 234 nM T62460 CDTG10 155518349 IC50 = 4 nM T62460 CQ19HO 155518921 IC50 = 4 nM T62460 CLK4S9 155519594 IC50 = 1510 nM T62460 CF0H9V 155520176 IC50 = 124 nM T62460 C0A9LX 155520276 IC50 > 10000 nM T62460 C4YJN9 155520341 IC50 = 17 nM T62460 C1PJC7 155520619 IC50 = 130 nM T62460 C0YEX7 155521332 IC50 = 38 nM T62460 CXG4L3 155522806 IC50 = 3.4 nM T62460 C9LUO3 155523352 IC50 = 43 nM T62460 C7NVQ5 155523535 IC50 = 380.2 nM T62460 C32POG 155523862 IC50 = 996.2 nM T62460 CE4FX7 155525956 IC50 = 469.2 nM T62460 CCS24O 155527492 IC50 = 2630.4 nM T62460 CK14UT 155528172 IC50 = 748 nM T62460 CB26JT 155528364 IC50 = 33 nM T62460 CVW07K 155528897 IC50 = 121 nM T62460 CL47NH 155529550 IC50 = 180 nM T62460 CRX08F 155531665 IC50 = 260 nM T62460 CQU09F 155532106 IC50 = 27 nM T62460 C5V6PY 155532206 IC50 > 2000 nM T62460 C4LE7Q 155532724 IC50 = 23 nM T62460 CLSV71 155533995 IC50 = 110 nM T62460 CGH63O 155534464 IC50 = 1.9 nM T62460 C2NPE6 155534808 IC50 = 110 nM T62460 C64FIW 155534972 IC50 = 842 nM T62460 CE8QW2 155535975 IC50 = 13 nM T62460 CMV7B2 155538485 IC50 = 2400 nM T62460 C5GNH8 155538704 IC50 = 285 nM T62460 C5WB0T 155539358 IC50 = 9670 nM T62460 C03BNT 155539537 IC50 = 10800 nM T62460 C3O6KI 155540160 IC50 = 92 nM T62460 C0D8OL 155540191 IC50 = 28.84 nM T62460 C16MHE 155540242 IC50 > 2000 nM T62460 CBA08W 155540345 IC50 = 11500 nM T62460 CP2NY0 155540484 IC50 = 4.169 nM T62460 CF8O5T 155540488 IC50 = 831.76 nM T62460 C51JNT 155540621 IC50 = 5.495 nM T62460 C76QBR 155541045 IC50 = 2200 nM T62460 CT1AX5 155541077 IC50 = 6.918 nM T62460 CY8F7S 155541097 IC50 = 104 nM T62460 CH6LV1 155541475 IC50 = 70.79 nM T62460 CS58BA 155541478 IC50 = 920 nM T62460 CF9AX3 155542099 IC50 = 750 nM T62460 C1B6EK 155542401 IC50 = 25.12 nM T62460 CH59RW 155542578 IC50 = 13 nM T62460 CKL31P 155542961 IC50 = 69.18 nM T62460 CH46TG 155543289 IC50 = 643 nM T62460 C1QRZ2 155543349 IC50 = 14 nM T62460 CKM8G4 155543489 IC50 = 1821 nM T62460 CRA21U 155543538 IC50 = 1159 nM T62460 CD9Z3W 155544141 IC50 = 8.7 nM T62460 CZ3YI6 155544372 IC50 = 943 nM T62460 CTQ63L 155544706 IC50 = 33.88 nM T62460 CP7XE1 155545114 IC50 = 29.51 nM T62460 CFR42U 155545338 IC50 = 104.71 nM T62460 C5BHW8 155546008 IC50 = 43 nM T62460 C5U8HP 155546232 IC50 = 37.15 nM T62460 CJ8F7V 155546474 IC50 = 33900 nM T62460 CSI1U9 155547916 IC50 = 81 nM T62460 C0B3RK 155547921 IC50 = 169.82 nM T62460 C3DZU0 155548345 IC50 = 40 nM T62460 CPR01A 155549631 IC50 = 2270 nM T62460 CI6Y5Z 155549690 IC50 = 3.981 nM T62460 C10OSG 155550219 IC50 = 40 nM T62460 C3DW8J 155550308 IC50 = 9.333 nM T62460 C31QUW 155550462 IC50 = 32 nM T62460 C6UJS7 155550600 IC50 = 200 nM T62460 C0DMP2 155551420 IC50 = 1240 nM T62460 CHM8G1 155551600 IC50 = 22000 nM T62460 C2Q1LR 155552255 IC50 = 20 nM T62460 CW1UX0 155552333 IC50 = 11.48 nM T62460 CV4NX3 155552736 IC50 = 7940 nM T62460 C62ERW 155552853 IC50 = 31.62 nM T62460 CPB6M8 155553409 IC50 = 923 nM T62460 C5HQ7X 155553551 IC50 = 6 nM T62460 CADO35 155554376 IC50 = 414 nM T62460 CNTP52 155554413 IC50 = 63 nM T62460 CWLC85 155554605 IC50 = 104 nM T62460 CQ6S8E 155554939 IC50 = 16.6 nM T62460 C47MNG 155554972 IC50 = 1100 nM T62460 CP39ZD 155555305 IC50 = 295.12 nM T62460 C9J4HM 155555486 IC50 = 3473 nM T62460 CTRV23 155555922 IC50 = 460 nM T62460 C2VS8X 155556321 IC50 = 1319 nM T62460 CG48UE 155556474 IC50 = 9.12 nM T62460 C8TYG7 155556520 IC50 > 9524 nM T62460 C59HKP 155557055 IC50 > 3000 nM T62460 CH9ON1 155557340 IC50 = 1242 nM T62460 CZUT98 155557375 IC50 = 460 nM T62460 CG9E7Z 155557901 IC50 = 151 nM T62460 CHW4O3 155558352 IC50 = 16.6 nM T62460 C7HFI8 155558403 IC50 = 47 nM T62460 C2LK9V 155558426 IC50 = 2032 nM T62460 C7WND0 155558729 IC50 = 199 nM T62460 C3V5HL 155559143 IC50 = 96.2 nM T62460 C2U5ZM 155559343 IC50 = 34.67 nM T62460 CSF54R 155559609 IC50 = 1262 nM T62460 CANJ25 155559746 IC50 = 851.14 nM T62460 C46KLS 155559780 IC50 > 1000 nM T62460 CNK81M 155560413 IC50 = 54.95 nM T62460 C54NQC 155561203 IC50 = 76 nM T62460 C1Z6IL 155561218 IC50 = 90 nM T62460 CH1LJ2 155562424 IC50 = 1586 nM T62460 CRU0K3 155563465 IC50 = 9290 nM T62460 C68TCL 155563799 IC50 = 774 nM T62460 C1NM2T 155564180 IC50 = 1820 nM T62460 CBQN81 155564466 IC50 = 1126 nM T62460 CZ2NK9 155565077 IC50 = 2884.03 nM T62460 CA0Z1U 155565486 IC50 = 21600 nM T62460 CSNF76 155565806 IC50 = 14.13 nM T62460 CF1X5I 155566525 IC50 = 122 nM T62460 C7S5MC 155566661 IC50 > 3000 nM T62460 CQA46B 155566981 IC50 = 10500 nM T62460 C6AXL1 155567447 IC50 = 2610 nM T62460 CSRZ04 155567801 IC50 > 3000 nM T62460 CGX28M 155567987 IC50 = 1700 nM T62460 COS7X5 155568028 IC50 = 253.8 nM T62460 COGC41 155568181 IC50 = 287.4 nM T62460 C0L6UT 155568261 IC50 = 19.05 nM T62460 CR79DJ 155568314 IC50 > 3000 nM T62460 C8EYW3 155568955 IC50 = 852 nM T62460 CRHE56 155569596 IC50 = 8800 nM T62460 CE50IC 155569626 IC50 = 3300 nM T62460 C3X6WU 155569641 IC50 = 764 nM T62460 C14DIR 16750188 IC50 = 3000 nM T62460 C5UI4F 16750189 IC50 = 5800 nM T62460 C6JKT9 16750206 IC50 > 10000 nM T62460 CYIU14 16750228 IC50 = 3500 nM T62460 CX4I6T 16750253 IC50 = 1700 nM T62460 CI79TY 16750254 IC50 = 8700 nM T62460 CS6UT4 16750288 IC50 = 3600 nM T62460 COM3C1 16750290 IC50 = 4600 nM T62460 CI67WG 16750292 IC50 = 1000 nM T62460 CIGJ63 16750308 IC50 = 3600 nM T62460 CL2SY5 16750330 IC50 = 4900 nM T62460 CE5P2I 53363072 IC50 = 2500 nM T62460 CTV60O 53363073 IC50 = 3100 nM T62460 CD74BW 53363074 IC50 = 2800 nM T62460 CU3M8P 53363075 IC50 > 10000 nM T62460 C07FTA 53363076 IC50 > 10000 nM T62460 C9JX2G 53363150 IC50 = 950 nM T62460 CJ04SF 53363151 IC50 = 1300 nM T62460 CO7Z2P 53363152 IC50 = 940 nM T62460 C1T2LY 53363154 IC50 = 2100 nM T62460 C9GEA7 53363242 IC50 = 2400 nM T62460 CTSP38 53363245 IC50 = 1900 nM T62460 CM7BZ3 53363246 IC50 = 830 nM T62460 C0QON7 53363337 IC50 = 380 nM T62460 CU76JB 53363338 IC50 > 10000 nM T62460 C2PU3M 53364335 IC50 > 10000 nM T62460 C10FXI 53364337 IC50 = 1900 nM T62460 C2U9QE 53364338 IC50 = 400 nM T62460 D02BXJ 46864270 IC50 = 55.3 nM T62460 D03BQI 3794 IC50 > 10000 nM T62460 D06HVH 54613583 IC50 > 10000 nM T62460 D09HVH 135566652 IC50 > 10 nM T62460 D0E5IP 3795 IC50 > 10000 nM T62460 D0H7DQ 6419755 IC50 = 770 nM T62460 D0IR6U 5494425 IC50 = 4 nM T62460 D0US9O 45275255 IC50 < 3 nM T62460 D0V6VQ 53344620 IC50 = 37.5 nM T62460 D0VC0I 5169 IC50 > 100000 nM T96014 D06TNL 3278 IC50 = 14000 nM T96014 D06ZAY 3561 IC50 = 500 nM T96014 D0Y2NE 448537 IC50 = 75000 nM T96014 D0B1FE 3194 IC50 = 14 nM T96014 C3MGF2 44419685 IC50 = 12000 nM T22274 D01QIN 60823 IC50 = 14466 nM T22274 D03RTS 2662 IC50 = 643 nM T22274 D04LKS 25126798 IC50 = 15 nM T22274 D06WTZ 53232 IC50 = 16285 nM T22274 D07POC 176870 IC50 > 32000 nM T22274 D08CDI 208908 IC50 > 10000 nM T22274 D0AZ3C 5291 IC50 > 100000 nM T22274 D0E3SH 6918837 Ki = 0.7 nM T22274 D0E7PQ 5311 Ki = 1 nM T22274 D0L7LC 5352062 Ki = 9.5 nM T22274 D0Y3KG 3121 IC50 > 2000000 nM T22274 D00FHR 9865515 IC50 > 10000 nM T22274 D00SSZ 11178958 IC50 = 1600 nM T22274 D01UXJ 11609955 IC50 = 72 nM T22274 D01WKZ 53340426 IC50 = 2.6 nM T22274 D05KED 53340666 IC50 = 4.7 nM T22274 D06TKI 49857317 IC50 = 2100 nM T22274 D07FPY 6918877 Ki = 20 nM T22274 D09XIZ 11538455 Ki = 16.9 nM T22274 D0B1FE 3194 IC50 = 1200 nM T22274 D0B3FV 6445533 IC50 = 5.93 nM T22274 D0B7CH 4775 IC50 = 240000 nM T22274 D0E6UZ 54575456 IC50 = 8 nM T22274 D0GH3Q 9804992 Ki = 4.2 nM T22274 D0L2UQ 49855250 Ki = 247 nM T22274 D0M8FD 4261 IC50 = 3930 nM T22274 D0V0SL 11749858 Ki = 17 nM T22274 D0XT6W 6918638 Ki = 1.6 nM T22274 D0Z4RC 24756910 IC50 = 5.1 nM T22274 D0J8OC 5186 Ki = 0.25 nM T22274 D00HXJ 118884610 Ki = 0.7 nM T22274 D0CH8Q 56965342 IC50 > 10000 nM T22274 D0JY1I 42613483 IC50 = 41 nM T22274 D0L1NO 72722126 IC50 = 3100 nM T22274 D0N2DK 72710871 IC50 = 2 nM T22274 D0Q1QY 57381425 IC50 = 1.7 nM T22274 D0QX3G 71532921 IC50 = 56 nM T22274 D0V5IQ 130227480 IC50 = 66 nM T22274 D0YN2T 86302836 IC50 = 6100 nM T22274 D0ZG5X 71811260 IC50 = 11 nM T22274 D0N3SH 4996 Ki = 4.8 nM T22274 D0W9NH 2746 IC50 > 40000 nM T22274 C8HA6K 3994 IC50 = 750 nM T22274 CBIR94 10313 IC50 = 115 nM T22274 CL25FN 76175 IC50 > 30000 nM T22274 C1N2KZ 88129 IC50 = 16000 nM T22274 C5Z1QA 96028 IC50 > 200000 nM T22274 CE42TU 119411 IC50 > 25000 nM T22274 CF60JA 220184 IC50 = 1100 nM T22274 CPZ3A5 245297 IC50 = 1395 nM T22274 CUD3X6 252888 IC50 = 65000 nM T22274 CCM91F 264313 IC50 > 720000 nM T22274 C35INR 338818 IC50 > 40000 nM T22274 CH1JD3 419176 IC50 = 2000 nM T22274 CG8E6F 443484 IC50 = 80000 nM T22274 C5PGB9 604917 IC50 = 300 nM T22274 C0Y4WC 614947 Ki > 2500 nM T22274 CAOM82 729359 IC50 = 320000 nM T22274 C3FA2Y 770976 IC50 = 180000 nM T22274 C0EM9B 801008 IC50 = 37400 nM T22274 CU3HS2 1108280 IC50 > 100000 nM T22274 CFZJ76 1187508 IC50 = 200000 nM T22274 CXLY12 1520179 IC50 = 45000 nM T22274 C96GFC 1798422 IC50 = 135900 nM T22274 C2PXB3 1973480 IC50 = 5100 nM T22274 CT08IQ 2378263 IC50 = 200000 nM T22274 CW76QZ 2385952 IC50 = 150000 nM T22274 CA9TW1 2723947 IC50 = 681 nM T22274 CW9CU3 3151732 IC50 = 100000 nM T22274 CK8I3T 3432579 IC50 = 376 nM T22274 CZA83Y 4118131 IC50 = 448 nM T22274 C53JHV 4245760 IC50 = 240000 nM T22274 CV9JS5 4288771 IC50 = 650 nM T22274 CBO4Y9 4961664 IC50 = 390000 nM T22274 CFQ23S 4962314 IC50 = 190000 nM T22274 CFKI56 4962437 IC50 = 51000 nM T22274 CFT78S 5111969 IC50 = 77000 nM T22274 CN4M6D 5281220 IC50 = 48500 nM T22274 CSIJ53 5793932 IC50 = 26900 nM T22274 C18ENP 6918846 Ki = 27 nM T22274 C1RD7E 6918878 IC50 > 10000 nM T22274 CX46OG 7130899 IC50 = 2300 nM T22274 CR3W8A 7131995 IC50 = 55000 nM T22274 CFUI51 8866284 IC50 = 6900 nM T22274 CJY6B3 9102265 IC50 = 44000 nM T22274 CP93LF 9533923 IC50 = 95000 nM T22274 CJ07ZA 9800555 IC50 = 7230 nM T22274 CAU23Y 9806551 IC50 = 40 nM T22274 CC0EU7 9828788 IC50 = 330 nM T22274 CH2LR4 9835152 IC50 = 7 nM T22274 CLYJ85 9848223 IC50 = 620 nM T22274 C4GBE9 9860473 IC50 = 100 nM T22274 CSW4Y1 9891541 IC50 = 780 nM T22274 C81EYJ 9923508 IC50 = 2.5 nM T22274 CQG4V8 9924543 IC50 = 2 nM T22274 COLN58 9965621 IC50 = 4 nM T22274 CDT7U0 9998313 IC50 = 50 nM T22274 CR98AV 9999602 IC50 = 200 nM T22274 CXA5J1 10068980 IC50 = 79 nM T22274 CVC3A9 10071120 IC50 = 1050 nM T22274 CCD3S6 10090483 IC50 = 63 nM T22274 CWA9R2 10135838 IC50 > 32000 nM T22274 CL4C9H 10154438 Ki = 135.9 nM T22274 CB2OV7 10266393 IC50 = 79 nM T22274 C7RC1E 10309899 IC50 = 66 nM T22274 C5S8XH 10340474 IC50 = 160 nM T22274 C1G9YS 10362929 IC50 = 100 nM T22274 CN5IT3 10381402 IC50 = 100 nM T22274 C9OU5F 10464879 Ki > 2500 nM T22274 CDY91S 10584105 Ki = 527 nM T22274 C3KT5X 10707192 IC50 = 448 nM T22274 CSMT47 10728039 Ki > 2500 nM T22274 C3FC7X 10800939 IC50 = 5360 nM T22274 CK8UV7 11019840 Ki > 2500 nM T22274 CW2GJ0 11166750 IC50 = 79 nM T22274 CFEN82 11177718 IC50 = 79 nM T22274 CMQ38G 11199235 IC50 = 120 nM T22274 C8G5WP 11210533 IC50 = 6500 nM T22274 CG27ZR 11212396 IC50 = 79 nM T22274 C89SVA 11223999 IC50 = 63 nM T22274 CYJ60V 11244651 IC50 = 800 nM T22274 CSO06H 11259022 IC50 = 63 nM T22274 CI7W3O 11267278 IC50 = 114 nM T22274 C6AKW1 11270791 IC50 = 79 nM T22274 CM6ZW2 11279156 IC50 = 482 nM T22274 CV9Y4T 11326181 IC50 = 160 nM T22274 CCT25X 11340446 IC50 = 107 nM T22274 CZT79Q 11360420 IC50 = 63 nM T22274 C9QB0C 11396478 IC50 = 63 nM T22274 CVH8N1 11430412 IC50 = 120 nM T22274 CRTV86 11430535 IC50 = 63 nM T22274 C5HP1B 11441977 IC50 = 50 nM T22274 CLW8E4 11477101 IC50 = 943 nM T22274 CB3N5M 11514394 IC50 = 37 nM T22274 CRZ7H2 11556677 IC50 = 680000 nM T22274 C2F9NT 11558827 IC50 = 34.5 nM T22274 C9UN7F 11637884 IC50 = 1500 nM T22274 C24SBP 11657529 IC50 = 120 nM T22274 CQ32FV 11664499 IC50 = 45 nM T22274 CG9OC4 11682502 IC50 = 224 nM T22274 CYB26W 11688197 IC50 = 24.4 nM T22274 CE4Z0Y 11844891 IC50 = 29 nM T22274 C6JF9E 11844892 IC50 = 36 nM T22274 CY0WV6 11844893 IC50 = 23 nM T22274 CU0M1E 11947684 IC50 = 9.1 nM T22274 CF06BI 11963978 IC50 = 881 nM T22274 C9G1BN 11993595 IC50 = 4900 nM T22274 CH5JS7 11993694 IC50 = 2.6 nM T22274 CJQ8L0 12001305 IC50 = 897 nM T22274 C1BVY9 12325934 IC50 > 30000 nM T22274 CKI97Z 12344252 IC50 > 200000 nM T22274 CKSL53 12507616 IC50 > 200000 nM T22274 CJ94OC 12542182 Ki > 2500 nM T22274 COF8W3 13008156 IC50 > 50000 nM T22274 C06UTF 13507024 IC50 = 22 nM T22274 CA07QT 13873842 IC50 > 50000 nM T22274 C1KR4L 14113324 IC50 > 50000 nM T22274 C15MQN 14113325 IC50 > 50000 nM T22274 C2D1KP 15983982 Ki = 300 nM T22274 CA2YF9 15984018 IC50 = 360 nM T22274 CHB82E 15986417 IC50 = 2800 nM T22274 C52EVH 15986418 IC50 = 41.8 nM T22274 CS1QO9 15986509 IC50 = 36.8 nM T22274 C5T1WF 16006672 IC50 > 10000 nM T22274 CQGC05 16036765 IC50 = 13 nM T22274 CM3T2E 16049824 IC50 = 10 nM T22274 CRL96K 16065840 IC50 = 190 nM T22274 C30UFT 16066811 IC50 > 50000 nM T22274 CFK8J5 16068056 Ki = 94 nM T22274 CMQP70 16068495 Ki = 225 nM T22274 CT84XO 16068594 Ki = 348 nM T22274 CF3ZG5 16068595 Ki = 282 nM T22274 CL60CA 16068912 Ki = 227 nM T22274 C9ZQB3 16095102 IC50 > 50000 nM T22274 C80XYC 16095113 IC50 > 50000 nM T22274 C6BGM2 16659535 IC50 = 40 nM T22274 CQI9N3 16659537 IC50 = 10 nM T22274 C5YFV9 16661453 IC50 = 310 nM T22274 C8S5OX 16661455 IC50 = 150 nM T22274 CH67WF 16661458 IC50 = 220 nM T22274 CZ72YC 16661613 IC50 = 10 nM T22274 C8DZ1T 16661615 IC50 = 40 nM T22274 CQV40I 16661617 IC50 = 50 nM T22274 C5CIB4 16663079 IC50 > 50000 nM T22274 CUG50I 16733294 IC50 = 7.5 nM T22274 CWO7V0 16733295 IC50 = 73 nM T22274 C4W0PG 16733410 IC50 = 5.4 nM T22274 C0MO3Z 16733411 IC50 = 3.7 nM T22274 C3QL4X 16733412 IC50 = 620 nM T22274 CV54SY 16733414 IC50 = 21 nM T22274 C1VCX2 16733415 IC50 = 45.5 nM T22274 CXN07K 16733416 IC50 = 2010 nM T22274 CP9AR8 16733417 IC50 = 9 nM T22274 CUE62T 16733590 IC50 = 216 nM T22274 CB4IN2 16773791 IC50 > 20000 nM T22274 C0ZWD2 17747368 IC50 = 1350 nM T22274 CS3PJ9 17747369 IC50 = 210 nM T22274 CKM7F9 17747371 EC50 = 640 nM T22274 CQHD27 20459443 IC50 = 12 nM T22274 C2X5PQ 22958841 EC50 = 19200 nM T22274 CEF8W4 23625604 IC50 = 1220 nM T22274 C5RO8F 23625605 IC50 = 180 nM T22274 CQ12UX 23626081 IC50 = 280 nM T22274 C70BKU 23640756 IC50 = 1690 nM T22274 CB8A5Q 23648260 IC50 > 50000 nM T22274 C36NKL 23648268 IC50 > 20000 nM T22274 CS9WX8 23649315 IC50 = 230 nM T22274 CH35NV 23656767 IC50 > 10000 nM T22274 CE85CP 23657268 IC50 = 4922 nM T22274 CU01QJ 24178404 IC50 = 3 nM T22274 C4UV3T 24726843 IC50 = 550 nM T22274 C5G7IV 24726844 IC50 = 550 nM T22274 C8RC9P 24744325 IC50 > 50000 nM T22274 C17GDO 24779722 IC50 = 20.1 nM T22274 CY12VH 24825455 Ki = 28 nM T22274 CIO7Q6 24853792 IC50 = 970 nM T22274 CBN0J5 24853793 IC50 = 340 nM T22274 CI3B6L 24857909 IC50 = 89 nM T22274 CLT5J2 24881257 IC50 = 4.8 nM T22274 C5GCM1 24881328 IC50 = 1.9 nM T22274 C8QVB1 24881329 IC50 = 4.4 nM T22274 CU0AM3 24881330 IC50 = 3.1 nM T22274 CQM51L 24881331 IC50 = 9.6 nM T22274 C4KH8F 24881332 IC50 = 7.3 nM T22274 C1KA3V 24881333 IC50 = 4.2 nM T22274 C47APB 24881402 IC50 = 3.3 nM T22274 CSN8W1 24881403 IC50 = 7.5 nM T22274 C1UQ3K 24881404 IC50 = 1.3 nM T22274 C51TMH 24881405 IC50 = 2.6 nM T22274 C9EZI7 24881406 IC50 = 1.9 nM T22274 C6P3HS 24881407 IC50 = 3.1 nM T22274 CZ3TU1 24881464 IC50 = 3.5 nM T22274 CDI49N 24881465 IC50 = 3.8 nM T22274 CQGP87 24881466 IC50 = 2.8 nM T22274 CQC8T7 24882475 IC50 = 4900 nM T22274 CS1MH8 24888322 IC50 > 30000 nM T22274 CPU1Z5 24893969 IC50 = 43 nM T22274 CP29ZE 24893970 IC50 = 65 nM T22274 CHKZ02 24894417 IC50 = 110 nM T22274 C6BNX7 24894418 IC50 = 132 nM T22274 CQ63WU 24894419 IC50 = 1640 nM T22274 C3E0SN 24894423 IC50 = 329 nM T22274 CA56SQ 24894517 IC50 = 346 nM T22274 CVA4J1 24894518 IC50 = 23 nM T22274 C7FV6W 24894519 IC50 = 90 nM T22274 C8R2KN 24894520 IC50 = 256 nM T22274 CO2XH9 24894521 Ki = 140 nM T22274 C2EQS1 24894522 IC50 = 517 nM T22274 CJWI39 24894523 IC50 = 521 nM T22274 CJ15OF 24894524 IC50 = 175 nM T22274 CKQZ25 24894639 IC50 = 382 nM T22274 CITS83 24894640 IC50 = 38 nM T22274 CX3QD8 24894641 IC50 = 421 nM T22274 CC1G2E 24894642 IC50 = 119 nM T22274 CJ64TA 24894643 IC50 = 830 nM T22274 C1PTW8 24894644 IC50 = 198 nM T22274 CKJC01 24894645 IC50 = 483 nM T22274 CW3MP6 24894775 IC50 = 1450 nM T22274 C6YL4C 24894776 IC50 = 979 nM T22274 CA2O6T 24894777 IC50 = 245 nM T22274 C8XS0N 24894778 IC50 = 519 nM T22274 C6CK9N 24894779 IC50 = 181 nM T22274 CXY5C7 24894780 IC50 = 44 nM T22274 CT4RJ0 24894895 IC50 = 396 nM T22274 CJTP74 24894896 IC50 = 250 nM T22274 C4F5TN 24894897 IC50 = 116 nM T22274 C75WEJ 24894898 IC50 = 390 nM T22274 CMT7F4 24894899 IC50 = 89 nM T22274 CH13WV 24894900 IC50 = 195 nM T22274 CA5V7S 24894901 IC50 = 301 nM T22274 CDU08E 24895004 IC50 = 606 nM T22274 C1IR2A 24895005 IC50 = 340 nM T22274 CQJ78L 24895006 IC50 = 1250 nM T22274 C4PN6I 24895007 IC50 = 2040 nM T22274 C9H1WI 24895008 IC50 = 431 nM T22274 CYM91Q 24895009 IC50 = 135 nM T22274 CEH9A4 24895010 IC50 = 245 nM T22274 C8SP7C 24895115 IC50 = 175 nM T22274 C0C9VU 24895116 IC50 = 204 nM T22274 CM3Q7A 24895117 IC50 = 438 nM T22274 CZ1SP9 24895118 IC50 = 94 nM T22274 CY7D1N 24895120 IC50 = 4570 nM T22274 CH7L8Z 24895121 IC50 = 2130 nM T22274 C60FAX 24895122 IC50 = 18 nM T22274 CO68DV 24895187 IC50 = 816 nM T22274 C40QJO 24895188 IC50 = 1090 nM T22274 C2K8BR 24895189 IC50 = 102 nM T22274 CBI25A 24895190 IC50 = 104 nM T22274 C73LSX 24896624 EC50 = 1000 nM T22274 CC0R9O 24938735 IC50 = 28.11 nM T22274 CF03HD 24948905 IC50 = 31.6 nM T22274 CHP8O6 24948906 IC50 = 2.54 nM T22274 C1KRT8 24948907 IC50 = 72.2 nM T22274 CKY2P8 24948908 IC50 = 5.86 nM T22274 C25CFI 24948909 IC50 = 35.1 nM T22274 CWQ04Z 24948910 IC50 = 6.81 nM T22274 CM9I3X 24951310 IC50 = 49.5 nM T22274 CX1YF8 24951311 IC50 = 61.9 nM T22274 CV10XU 24951312 IC50 < 0.002 nM T22274 CD6KV0 24951313 IC50 = 3.98 nM T22274 CQY9Z0 24951314 IC50 = 0.326 nM T22274 C5B0IJ 25023793 IC50 = 1700 nM T22274 CHE82I 25023795 IC50 = 310 nM T22274 CX8G3W 25023796 IC50 = 210 nM T22274 CVRS37 25023797 IC50 = 230 nM T22274 C7GO3U 25023798 IC50 = 150 nM T22274 C3G2AU 25023799 IC50 = 240 nM T22274 CAS18V 25023800 IC50 = 460 nM T22274 CX7D5B 25023801 IC50 = 130 nM T22274 CZG50I 25023802 IC50 = 310 nM T22274 CF9WH6 25023808 IC50 = 15 nM T22274 CVS1M4 25023811 IC50 = 490 nM T22274 C2O9CE 25023812 IC50 = 840 nM T22274 CW6KR2 25023813 IC50 = 410 nM T22274 C10CNP 25023814 IC50 = 2500 nM T22274 C5IJ6X 25023815 IC50 = 730 nM T22274 C24MTU 25023816 IC50 = 640 nM T22274 CKY94C 25023817 IC50 = 2000 nM T22274 CJG8C5 25023818 IC50 = 1300 nM T22274 CLA50V 25023819 IC50 = 1500 nM T22274 C86TAU 25023820 IC50 = 580 nM T22274 CTC0H5 25023821 IC50 = 4200 nM T22274 CHX6A5 25023822 IC50 = 2500 nM T22274 CV8EF6 25032862 IC50 > 50000 nM T22274 CX69SY 25066355 IC50 = 15.6 nM T22274 CF8VP4 25066356 IC50 = 10.1 nM T22274 CS9XH7 25066547 IC50 = 9.38 nM T22274 C46AGN 25066548 IC50 = 1.97 nM T22274 CJF2M7 25066549 IC50 = 8.44 nM T22274 C9X0JM 25099146 IC50 = 690 nM T22274 CJ41EF 25099147 IC50 = 9990 nM T22274 CPTI96 25110599 IC50 = 800 nM T22274 CY9JV6 25113671 IC50 = 148.5 nM T22274 C7ZN2W 25118059 IC50 = 0.6 nM T22274 CGW49I 25146686 IC50 > 200000 nM T22274 C4GC5R 25151496 IC50 = 78 nM T22274 CFO6B0 25151497 IC50 = 117.4 nM T22274 CTP21Q 25151864 IC50 = 89.3 nM T22274 C4I1CJ 25155417 IC50 > 50000 nM T22274 CB4E2J 25155956 IC50 > 50000 nM T22274 CFS5O4 25168576 IC50 = 650 nM T22274 C0R5OK 25168856 IC50 = 240 nM T22274 CO14XG 25195084 IC50 > 20000 nM T22274 CE5F2V 25195975 IC50 = 20 nM T22274 C6BDX3 25207860 IC50 = 81000 nM T22274 CB29PE 25211681 IC50 = 180 nM T22274 CM57WO 25211776 IC50 = 3350 nM T22274 CU25TK 25211878 IC50 = 60 nM T22274 C2YG9N 25216677 IC50 = 4100 nM T22274 C5CZV0 25216678 IC50 = 250 nM T22274 CB6C2A 25216810 IC50 = 450 nM T22274 CPX03T 25217055 IC50 = 1700 nM T22274 CP26WM 25217056 IC50 = 1800 nM T22274 CBDR02 25217057 IC50 = 100 nM T22274 C9URH7 25217288 IC50 = 320 nM T22274 C2WH9J 25217398 IC50 = 2000 nM T22274 CSM0F2 25217513 IC50 = 890 nM T22274 C5FZ2V 25225123 IC50 = 4010 nM T22274 CCD5M7 25227504 IC50 = 0.84 nM T22274 CK0D5S 25227505 IC50 = 10.2 nM T22274 CN97JP 25227508 IC50 = 3.43 nM T22274 CW8R1B 25227513 IC50 = 3.92 nM T22274 CPNQ02 25257992 IC50 > 30000 nM T22274 CE0NV4 25257993 IC50 = 48.55 nM T22274 C43BHY 25269097 IC50 = 27 nM T22274 CN7K1S 25374100 IC50 = 1300 nM T22274 C3XVL1 40173316 IC50 = 25000 nM T22274 CU53WB 42596953 IC50 = 86 nM T22274 CJ1RQ7 42598706 IC50 = 25 nM T22274 C2LES7 42599455 IC50 = 3.5 nM T22274 C2KO0F 42599456 IC50 = 3.4 nM T22274 C1UAO7 42601485 IC50 > 50000 nM T22274 C3P6NY 42601488 IC50 = 480 nM T22274 COI7Y3 42611300 IC50 > 10000 nM T22274 CU23PG 42611301 IC50 = 31 nM T22274 C3ZV9H 42611302 IC50 = 2700 nM T22274 CW1G2R 42611390 IC50 > 10000 nM T22274 C62QFJ 42611486 IC50 > 10000 nM T22274 CQ37HN 42612743 IC50 = 102 nM T22274 CLH2Q7 42612852 IC50 = 2310 nM T22274 C7GIQ3 42625508 IC50 = 36 nM T22274 CVZ83M 42625582 IC50 >= 32000 nM T22274 C5MD9E 42625892 IC50 > 100000 nM T22274 CDT65Y 42631047 IC50 = 3260 nM T22274 CB79DG 42637299 IC50 = 1100 nM T22274 CP36KB 42637300 IC50 = 24000 nM T22274 CI8J6H 42637372 IC50 = 110 nM T22274 C5RYO0 42637373 IC50 = 5600 nM T22274 CJ0CG5 42638004 IC50 = 14000 nM T22274 C8X0TG 42638005 IC50 = 320 nM T22274 C3LHF9 42917485 IC50 = 3600 nM T22274 CO57GS 44138033 IC50 = 94 nM T22274 CW4IX9 44178888 IC50 > 10000 nM T22274 C7RCY4 44178890 IC50 = 6100 nM T22274 CQ2VD5 44219634 IC50 = 82 nM T22274 CY0QB9 44253226 IC50 = 25.7 nM T22274 CZ8R1N 44253780 IC50 = 110 nM T22274 C6M5XJ 44268300 EC50 = 524000 nM T22274 C86IOC 44328927 IC50 > 10000 nM T22274 C7G5CO 44359547 IC50 = 910 nM T22274 CIT7A9 44359548 IC50 = 30000 nM T22274 CUM0Q6 44359555 IC50 = 3100 nM T22274 CP92JV 44359673 IC50 > 100000 nM T22274 CQ7J2G 44359674 IC50 = 5500 nM T22274 C2V4DN 44359681 IC50 = 600 nM T22274 CX31TB 44359788 IC50 = 2800 nM T22274 CQ5Y8G 44359800 IC50 > 100000 nM T22274 CL82CH 44359814 IC50 > 100000 nM T22274 CWY06M 44363182 EC50 = 19000 nM T22274 CN91KP 44363187 EC50 = 360000 nM T22274 C6ENC3 44427332 IC50 = 1250 nM T22274 C5YRC9 44431499 IC50 = 1500 nM T22274 C3U8EF 44442437 IC50 = 990 nM T22274 C9ZUW5 44442438 IC50 = 750 nM T22274 CJ6SN4 44442439 IC50 = 15000 nM T22274 CP71RI 44445956 IC50 = 280 nM T22274 C3KLP5 44445957 IC50 = 310 nM T22274 CF9RX6 44445958 IC50 = 230 nM T22274 CV7P0C 44447120 IC50 > 50000 nM T22274 CNC51G 44447194 IC50 > 50000 nM T22274 C5K7LA 44449588 Ki = 6.6 nM T22274 C90YQD 44452393 IC50 = 4670 nM T22274 COW2C1 44452422 IC50 = 1050 nM T22274 CAY46N 44452443 IC50 = 1130 nM T22274 CWRM21 44452444 IC50 = 2850 nM T22274 CRP6H9 44452468 IC50 = 1170 nM T22274 CN2GF3 44452469 IC50 = 2330 nM T22274 C9FL6O 44452486 IC50 = 4490 nM T22274 C0HP2A 44452501 IC50 = 1770 nM T22274 C0HR3Q 44452526 IC50 = 4020 nM T22274 CUO4I3 44452552 IC50 = 14720 nM T22274 C78CAQ 44452557 IC50 = 4090 nM T22274 CYBU71 44452577 IC50 = 2330 nM T22274 C8WKU9 44453790 IC50 = 98 nM T22274 C5VP4D 44454144 IC50 > 50000 nM T22274 C8A1ZD 44456564 IC50 = 15 nM T22274 CJ0L4C 44456965 IC50 = 13 nM T22274 C92UDN 44541230 IC50 = 6300 nM T22274 C7IB2P 44541231 IC50 = 29 nM T22274 C4TGM5 44541232 IC50 = 27 nM T22274 CR7W5C 44541233 IC50 > 1000 nM T22274 CFXD49 44541234 IC50 > 5000 nM T22274 C4FKU6 44541235 IC50 = 520 nM T22274 CE52NP 44543401 IC50 = 1900 nM T22274 CQI7O3 44543402 IC50 = 170 nM T22274 CJ0KH8 44543403 IC50 = 3100 nM T22274 C7H4FD 44543404 IC50 = 41 nM T22274 CGS14Q 44543405 IC50 = 15 nM T22274 CHX48R 44543406 IC50 = 37 nM T22274 CG2AE4 44543407 IC50 > 1000 nM T22274 C7F8YJ 44543715 Ki = 30 nM T22274 CW4KH2 44551271 IC50 = 14700 nM T22274 CW42BX 44562604 IC50 = 860 nM T22274 CDW54Z 44562605 IC50 = 600 nM T22274 C1WY8L 44562606 IC50 = 670 nM T22274 C9MB4K 44562607 IC50 = 160 nM T22274 CH2NP3 44562608 IC50 = 680 nM T22274 CBYZ26 44562609 IC50 = 2450 nM T22274 CZU3I7 44562657 IC50 = 11000 nM T22274 C3QSI4 44562762 IC50 = 270 nM T22274 CRJS52 44562763 IC50 = 580 nM T22274 C2LH1N 44562764 IC50 = 3000 nM T22274 CJ5US8 44562765 IC50 = 3540 nM T22274 CUT7L8 44562766 IC50 = 500 nM T22274 CH2KM0 44562767 IC50 = 840 nM T22274 CQX1R2 44562798 IC50 = 570 nM T22274 CQ5RJ3 44562799 IC50 = 170 nM T22274 C96LVR 44562800 IC50 = 710 nM T22274 CDY0E1 44562801 IC50 = 410 nM T22274 CEM91G 44562802 IC50 = 280 nM T22274 CEA9D0 44562840 IC50 = 700 nM T22274 C3DMN0 44563197 IC50 = 370 nM T22274 CGF8R5 44563236 IC50 = 580 nM T22274 CT63QG 44563237 IC50 = 330 nM T22274 CIO34V 44564642 Ki = 23 nM T22274 CTUG48 44568433 IC50 = 165 nM T22274 CG9OD1 44571302 IC50 = 10 nM T22274 C0ZX1A 44571330 IC50 = 170 nM T22274 CY83MO 44571331 IC50 = 110 nM T22274 CP6D1G 44571332 IC50 = 160 nM T22274 CUO3V0 44572289 IC50 = 200 nM T22274 CFH95O 44572348 IC50 = 600 nM T22274 CD17KA 44572349 IC50 = 190 nM T22274 CU4VC9 44572350 IC50 = 840 nM T22274 C5TBI9 44572351 IC50 = 280 nM T22274 COM65J 44572384 IC50 > 100000 nM T22274 CV91YE 44572385 IC50 > 100000 nM T22274 CAUH07 44572405 IC50 = 580 nM T22274 CUO41X 44572406 IC50 = 200 nM T22274 CY0I4X 44572407 IC50 = 420 nM T22274 C3CB2K 44572429 IC50 > 100000 nM T22274 CM2Q8J 44572430 IC50 > 100000 nM T22274 CAN4B0 44572431 IC50 >= 32000 nM T22274 C8AO6P 44572466 IC50 = 1400 nM T22274 C2O3IS 44572467 IC50 = 1100 nM T22274 CH09QJ 44572468 IC50 = 530 nM T22274 CMAT21 44572489 IC50 > 32000 nM T22274 CU1SY9 44572490 IC50 = 20900 nM T22274 CSD74G 44572491 IC50 > 100000 nM T22274 CZ2X7L 44572516 IC50 = 150 nM T22274 CW7BK3 44572517 IC50 = 560 nM T22274 C59TVW 44572518 IC50 = 370 nM T22274 CC74WS 44572519 IC50 = 520 nM T22274 CA9WO3 44572537 IC50 > 100000 nM T22274 C06SLW 44572538 IC50 > 100000 nM T22274 CY8TG3 44572539 IC50 > 100000 nM T22274 C1JR4C 44572540 IC50 = 91 nM T22274 CV50NO 44572558 IC50 = 1200 nM T22274 CB9Z4E 44572559 IC50 = 1200 nM T22274 C0RUB9 44572560 IC50 = 400 nM T22274 CY78SZ 44572561 IC50 = 480 nM T22274 CZ0PA9 44572581 IC50 = 89 nM T22274 CD9VR5 44572582 IC50 = 55 nM T22274 CG5UK0 44572584 IC50 = 45 nM T22274 CMX32U 44572633 IC50 = 39 nM T22274 CA3UR6 44572654 IC50 = 410 nM T22274 CMA3R6 44574139 IC50 = 68 nM T22274 C5KLR7 44574177 IC50 > 30000 nM T22274 CFS49I 44574178 IC50 > 30000 nM T22274 CJ32DK 44574179 IC50 > 30000 nM T22274 CQOS28 44574180 IC50 = 51 nM T22274 CN96ZV 44574181 IC50 = 885 nM T22274 CWJA85 44574206 IC50 = 17100 nM T22274 C46XHW 44574207 IC50 = 12300 nM T22274 C3RY9V 44574208 IC50 = 1710 nM T22274 CWKP93 44589698 IC50 = 170 nM T22274 CS4JP5 44589733 IC50 = 175 nM T22274 CEPG12 44589734 IC50 = 360 nM T22274 CZVO54 44589735 IC50 = 260 nM T22274 CPB1G7 44589736 IC50 = 160 nM T22274 CZ7VE6 44589745 IC50 = 1400 nM T22274 CDH14U 44589746 IC50 = 3500 nM T22274 CN18IR 44589774 IC50 = 410 nM T22274 CJMZ90 44589775 IC50 = 3320 nM T22274 C3O4NM 44591285 IC50 = 50000 nM T22274 CQ2WN9 44591286 IC50 > 10000 nM T22274 C8EK0X 44591287 IC50 > 10000 nM T22274 CNZ1M4 44591288 IC50 > 10000 nM T22274 CS6P3M 44591320 IC50 > 10000 nM T22274 CJI84H 44591321 IC50 > 10000 nM T22274 CV78HA 44591322 IC50 > 10000 nM T22274 C19IEO 44591323 IC50 > 10000 nM T22274 C18NCB 44591324 IC50 > 10000 nM T22274 C82VYI 44591343 IC50 = 440 nM T22274 CA6Q9Y 44592060 IC50 = 175 nM T22274 C0AC3P 44593559 IC50 = 900 nM T22274 CH2J8R 44598238 IC50 = 8000 nM T22274 CE5W3U 44598288 IC50 = 5800 nM T22274 C68BJH 44598289 IC50 = 3700 nM T22274 C9K2WV 44598290 IC50 = 7000 nM T22274 C16ZEP 44598291 IC50 > 10000 nM T22274 C28GHB 44598344 IC50 > 10000 nM T22274 CU65LR 44598345 IC50 = 1400 nM T22274 C41VTN 44598346 IC50 = 2320 nM T22274 CHQ86X 44598347 IC50 = 1080 nM T22274 CCVA51 44598385 IC50 = 4400 nM T22274 C29NXL 44598386 IC50 > 10000 nM T22274 C5WM7H 44598387 IC50 > 10000 nM T22274 CK8V9I 44598388 IC50 = 39 nM T22274 C2IS6D 44598428 IC50 > 10000 nM T22274 CJ54OH 44598429 IC50 = 70 nM T22274 C1TYW6 44598430 IC50 = 1120 nM T22274 C3TOK2 44598431 IC50 = 1670 nM T22274 CPZ65Q 44598479 IC50 > 10000 nM T22274 CGT51H 44598480 IC50 > 10000 nM T22274 CZ62IW 44598481 IC50 > 10000 nM T22274 C0OT6I 44598482 IC50 > 10000 nM T22274 CX8U6S 44598483 IC50 > 10000 nM T22274 CO5YJ8 44598535 IC50 = 4900 nM T22274 C5H8RA 44598536 IC50 > 10000 nM T22274 CC2QV9 44623002 IC50 = 4700 nM T22274 CVJ51M 44623152 IC50 > 50000 nM T22274 C6TJ2G 44623153 IC50 > 50000 nM T22274 C42SJP 45141750 IC50 = 22 nM T22274 CLE9U5 45141751 IC50 = 12 nM T22274 CL71OI 45483433 IC50 = 575 nM T22274 CUF94Q 45483434 IC50 = 716 nM T22274 C4S2PN 45483435 IC50 = 714 nM T22274 C02LVF 45485792 IC50 > 10000 nM T22274 C7EAV5 45485820 IC50 > 10000 nM T22274 CIO0T2 46179730 IC50 = 3.85 nM T22274 C2M4GV 46179732 IC50 = 3.3 nM T22274 CS75CD 46179779 IC50 = 3.1 nM T22274 C39YKM 46179780 IC50 = 4.3 nM T22274 C0CKE5 46180624 IC50 > 30000 nM T22274 C7GYH0 46180758 IC50 = 8.4 nM T22274 C27IKH 46180759 IC50 = 2.2 nM T22274 CSC1Y9 46180760 IC50 = 2.9 nM T22274 C4XHL5 46180761 IC50 = 1.7 nM T22274 C70FSJ 46180763 IC50 = 1.9 nM T22274 CD57RJ 46197798 IC50 = 118 nM T22274 CR04HA 46197799 IC50 = 110 nM T22274 C3ZE2B 46198177 IC50 = 457 nM T22274 CQ69AM 46205433 IC50 = 6 nM T22274 C7V1RE 46216758 IC50 = 330 nM T22274 CZ0F6R 46216759 IC50 = 410 nM T22274 C0RQ1B 46216760 IC50 = 280 nM T22274 CI06QG 46216772 IC50 = 240 nM T22274 C5U7GY 46230638 IC50 = 340 nM T22274 CN8F9S 46830326 IC50 = 79 nM T22274 C69UBY 46861822 IC50 = 2000 nM T22274 C8D4XL 46861823 IC50 = 24700 nM T22274 CB2G1W 46881144 IC50 = 7.6 nM T22274 C85RDN 46881213 IC50 = 2.52 nM T22274 CQTI31 46881225 IC50 > 30000 nM T22274 CM9W8B 46886948 IC50 = 63 nM T22274 C3X1PB 46886949 IC50 = 31 nM T22274 CA8ZB0 46886950 IC50 = 20 nM T22274 C5STW2 46887022 IC50 = 40 nM T22274 C35ATX 46887023 IC50 = 63 nM T22274 C35LCR 46887024 IC50 = 40 nM T22274 C1C7TX 46887025 IC50 = 79 nM T22274 CC6I4F 46887026 IC50 = 25 nM T22274 CEMV64 46887060 IC50 = 100 nM T22274 CCU65S 46887061 IC50 = 50 nM T22274 C24FTM 46887062 IC50 = 79 nM T22274 C8VD6Z 46887093 IC50 = 79 nM T22274 C3UNV6 46887094 IC50 = 63 nM T22274 CJE6Q2 46887127 IC50 = 100 nM T22274 C4OWH7 46887128 IC50 = 79 nM T22274 C74SPT 46887178 IC50 = 79 nM T22274 C9I6NF 46887179 IC50 = 79 nM T22274 C28RSA 46887180 IC50 = 100 nM T22274 CH85NX 46887211 IC50 = 63 nM T22274 C8YAV5 46887212 IC50 = 100 nM T22274 CJ30VB 46887241 IC50 = 120 nM T22274 CX53HE 46887282 IC50 = 400 nM T22274 CU38FK 46887283 IC50 = 630 nM T22274 C0CTM9 46887332 IC50 = 500 nM T22274 CP4W7O 46887556 IC50 = 25 nM T22274 C2GP9T 46887557 IC50 = 79 nM T22274 C3UIY6 46887558 IC50 = 79 nM T22274 CUR2X5 46887559 IC50 = 100 nM T22274 CMU9D7 46887584 IC50 = 40 nM T22274 CA8JT1 46887585 IC50 = 63 nM T22274 C25DSY 46887918 IC50 = 9400 nM T22274 C93CLK 46887919 IC50 = 33600 nM T22274 CPSI47 46890583 Ki = 8 nM T22274 C90NYX 46896338 IC50 > 30000 nM T22274 CU7L5W 46906597 IC50 = 50400 nM T22274 CG46KJ 46906641 IC50 = 31600 nM T22274 CAT34L 46906643 IC50 = 64000 nM T22274 C4V7PG 46907052 IC50 = 580 nM T22274 CSNU34 46907053 IC50 = 9300 nM T22274 CMQ3R0 46907054 IC50 = 3000 nM T22274 C05KTS 46907124 IC50 = 330000 nM T22274 C2PC1Z 46907160 IC50 = 1750 nM T22274 C72BEW 46907196 IC50 = 71300 nM T22274 C4V3ZK 46907197 IC50 = 191000 nM T22274 C6TRS7 46907198 IC50 = 153000 nM T22274 C0K4DL 46907280 IC50 = 101000 nM T22274 C3NE0Q 46907281 IC50 = 293000 nM T22274 C1HV6U 46907409 IC50 > 20000 nM T22274 CY7B1U 46913905 IC50 = 1916.9 nM T22274 C42UBP 46913906 IC50 = 3203.1 nM T22274 CWA0M8 46916092 IC50 = 1180.1 nM T22274 CYN9W5 46916093 IC50 = 728.7 nM T22274 C78XOJ 46916094 IC50 = 1709.8 nM T22274 C43TPV 46918824 IC50 = 39.81 nM T22274 CXH64A 46918825 IC50 = 1.4 nM T22274 C6GY9I 46934544 IC50 = 430 nM T22274 C3OD2Y 46934546 IC50 = 760 nM T22274 CL7PS1 49831258 IC50 = 36 nM T22274 C0OQX9 49831259 IC50 = 35 nM T22274 CI5L2P 49846123 IC50 = 51.25 nM T22274 C4DL0M 49847150 IC50 = 2.46 nM T22274 CC7Y9U 49850262 Ki = 3.3 nM T22274 C50PXU 49855444 IC50 = 430 nM T22274 CE7D2J 49855568 IC50 = 230 nM T22274 CFD9P3 49855569 IC50 = 1200 nM T22274 C1AU5N 49855758 IC50 = 230 nM T22274 CIFK93 49855759 IC50 > 10000 nM T22274 CK48OJ 49855760 IC50 > 10000 nM T22274 CZI3M1 49855761 IC50 > 32000 nM T22274 C9AVM0 49855833 IC50 = 130 nM T22274 CRPZ58 49855949 IC50 > 32000 nM T22274 CTU0K3 49855950 IC50 > 32000 nM T22274 CF85NL 49855951 IC50 > 32000 nM T22274 CF7YS9 49855952 IC50 = 9800 nM T22274 CJU38G 49855953 IC50 = 50 nM T22274 C6POK9 49856931 IC50 = 3300 nM T22274 CWM2L5 49871831 IC50 = 18 nM T22274 C1EOM0 49873200 IC50 = 20 nM T22274 CUFA67 50898589 IC50 = 0.704 nM T22274 CPOL89 50898669 IC50 = 2.96 nM T22274 CRHI06 50898670 IC50 = 3.05 nM T22274 CL7X3K 50898671 IC50 = 79.43 nM T22274 C5HPL0 50898672 IC50 = 0.972 nM T22274 CC1D9T 50898753 IC50 = 2.25 nM T22274 CC8F0Y 50898754 IC50 = 6.56 nM T22274 CZT96S 50898755 IC50 = 0.582 nM T22274 C6UOH5 50898756 IC50 = 0.459 nM T22274 CB75JS 50898757 IC50 = 2.99 nM T22274 C9A7XU 50898841 IC50 = 0.799 nM T22274 CQ43IF 50898842 IC50 = 8.96 nM T22274 CF0TI2 50898843 IC50 = 4.06 nM T22274 CJ1YC2 50898949 IC50 = 38.4 nM T22274 CKD7X9 50898950 IC50 = 11.5 nM T22274 C9BYZ1 50899047 IC50 = 4.9 nM T22274 CB89VJ 50899050 IC50 = 0.872 nM T22274 C59RDT 50899051 IC50 = 2.49 nM T22274 CPQ0F7 50991199 IC50 = 280 nM T22274 CV3X4J 51033161 IC50 > 50000 nM T22274 COA5W3 51051073 IC50 = 123 nM T22274 C5LZ4R 51351536 IC50 > 30000 nM T22274 CV76KB 51357270 IC50 = 151 nM T22274 CB87KG 52903573 IC50 = 350000 nM T22274 CVLE09 52950031 IC50 = 240 nM T22274 CYU0R2 52951254 IC50 = 141 nM T22274 C78BHS 52951255 IC50 = 116 nM T22274 C08BSF 52951359 IC50 = 164 nM T22274 CNC9V0 52951361 IC50 = 191 nM T22274 CSX0H2 52951363 IC50 = 163 nM T22274 C2IXJ1 52951365 IC50 = 169 nM T22274 CSB58V 52951464 IC50 = 94 nM T22274 CZ9FU4 52951465 IC50 = 158 nM T22274 C6DAB7 52952491 IC50 = 47 nM T22274 CO7B2Y 53239053 IC50 = 160 nM T22274 CE43FC 53249967 IC50 > 30000 nM T22274 C8SUQ5 53317424 IC50 > 30000 nM T22274 C7MO2J 53325871 IC50 = 3.3 nM T22274 CVM4Q3 53357987 IC50 = 30000 nM T22274 C78GKN 53361474 IC50 = 274 nM T22274 CNB63X 53361475 IC50 = 47 nM T22274 CQ43VH 53363518 Ki = 4 nM T22274 C6Y2EV 53374826 IC50 = 183 nM T22274 C86MWA 53380600 IC50 = 30400 nM T22274 CC5K2U 53380601 IC50 = 730 nM T22274 CN17BX 53380699 IC50 = 2250 nM T22274 C9WL1R 53387509 IC50 = 56 nM T22274 C2Y8VC 53390842 IC50 = 2100 nM T22274 C9U7GF 53464577 IC50 = 1 nM T22274 C4EYP7 53464578 IC50 = 3.3 nM T22274 C0WNH9 53464579 IC50 = 59.2 nM T22274 C4MQ3U 53464638 IC50 = 45.4 nM T22274 CJ53ZV 53464639 IC50 = 40.4 nM T22274 CN9RH2 53464770 IC50 = 18.3 nM T22274 CYQV72 54030066 IC50 = 4900 nM T22274 C0ZK7I 54576529 IC50 = 14.16 nM T22274 CTP2S1 54576530 IC50 = 15.93 nM T22274 CS8HY5 54576744 IC50 = 15.24 nM T22274 C5A7MU 54613496 IC50 = 1.9 nM T22274 CVP16C 54753629 IC50 = 8000 nM T22274 CQ1EX7 54770442 IC50 = 39.97 nM T22274 C7OJ4K 56602459 IC50 = 9900 nM T22274 CSY2L7 56602461 IC50 = 380 nM T22274 CIO96M 56659403 IC50 > 100000 nM T22274 CT4ZY0 56661203 IC50 = 230 nM T22274 C7R9TZ 56663191 IC50 = 35 nM T22274 CL18NI 56666337 IC50 > 100000 nM T22274 C9LC5Y 56673234 IC50 > 100000 nM T22274 CWH5N4 56673261 IC50 > 100000 nM T22274 C0ZJG3 56676500 IC50 = 1190 nM T22274 CFUT54 56682413 IC50 = 610 nM T22274 CQIL12 56755438 IC50 = 640000 nM T22274 C2ML5S 56837168 IC50 = 1.61 nM T22274 CCW89V 56932477 IC50 = 0.323 nM T22274 CGTC19 56932603 EC50 = 12450 nM T22274 CXU7E3 56932649 EC50 = 460 nM T22274 CX9I6N 56932650 EC50 = 5000 nM T22274 CIO27B 56932652 EC50 = 730 nM T22274 C6YH4J 56932655 EC50 = 1310 nM T22274 CXCF39 56932696 EC50 = 8700 nM T22274 C0FE5J 56932697 EC50 = 4950 nM T22274 C5XS1K 56932904 EC50 = 2250 nM T22274 CP63DG 56932907 EC50 = 990 nM T22274 CQ6GP1 56932909 EC50 = 1720 nM T22274 C7ABK4 56933019 EC50 = 11800 nM T22274 CZ25SN 56935695 IC50 > 30000 nM T22274 CVHR15 56950025 IC50 = 34.7 nM T22274 CH7W3C 56950026 IC50 = 22.5 nM T22274 CLV69W 56950027 IC50 = 3.06 nM T22274 C05BNS 56950152 IC50 = 1.02 nM T22274 CV2X3N 56950154 IC50 = 1.44 nM T22274 C83UDV 56964457 IC50 = 20 nM T22274 C3LSF8 57325671 IC50 = 555 nM T22274 CAW53S 57325672 IC50 = 30 nM T22274 C9P8HJ 57325755 IC50 = 19 nM T22274 C6PU3K 57326321 IC50 > 50000 nM T22274 C8XVR0 57326322 IC50 = 9500 nM T22274 CJY09O 57326509 IC50 = 30000 nM T22274 CS0PH3 57326510 IC50 > 50000 nM T22274 CQN86X 57326511 IC50 = 9000 nM T22274 CT58WK 57326610 IC50 = 8000 nM T22274 CP5EU9 57326611 IC50 > 50000 nM T22274 CG7S8T 57326612 IC50 > 50000 nM T22274 C7UY5V 57326613 IC50 = 5000 nM T22274 CDTL85 57326614 IC50 > 50000 nM T22274 CY0XG3 57326709 IC50 = 1000 nM T22274 CG6Z2X 57326710 IC50 = 1000 nM T22274 C9V5KT 57326712 IC50 = 250 nM T22274 C4ME8Z 57326713 IC50 = 320 nM T22274 C3Y5LI 57326714 IC50 = 220 nM T22274 C5YQ3I 57326715 IC50 = 2700 nM T22274 CP4EL2 57328394 IC50 = 260 nM T22274 CP2UN3 57336514 IC50 = 15 nM T22274 C10DMC 57336560 Ki = 20000 nM T22274 C8FLE6 57382288 IC50 = 7.5 nM T22274 C5CRJ1 57412107 IC50 = 190 nM T22274 COG4Q8 57412108 IC50 = 138 nM T22274 C3GAW0 57523757 EC50 = 2000 nM T22274 CBZV06 57523759 EC50 = 1100 nM T22274 C8CQ7V 57523845 IC50 = 240 nM T22274 C4SK5V 57524018 EC50 = 2600 nM T22274 CFHU47 57524021 IC50 = 21 nM T22274 CBZX29 57524107 EC50 = 360 nM T22274 C5LBS0 57524273 IC50 = 860 nM T22274 CVU30I 57524661 IC50 = 2260 nM T22274 CBM30D 57524665 EC50 = 6700 nM T22274 C3VU1R 57524666 EC50 = 2800 nM T22274 C3ZE4W 57524748 IC50 = 160 nM T22274 CJ68EZ 57524753 IC50 = 250 nM T22274 C4YNT9 57524833 IC50 = 140 nM T22274 C6A3CR 57524835 IC50 = 100 nM T22274 CTA82N 57524908 IC50 = 63 nM T22274 C46KFC 58147140 IC50 = 540 nM T22274 CA5Q6O 58147189 IC50 = 340 nM T22274 C3VLC7 58147195 IC50 = 340 nM T22274 C7TW0O 58147221 IC50 = 120 nM T22274 C4DYC0 58147224 IC50 = 560 nM T22274 CQS74A 58147262 IC50 = 580 nM T22274 C5E6RZ 58147291 IC50 = 490 nM T22274 CMP04X 58147302 IC50 = 260 nM T22274 CP8TZ4 58147401 IC50 = 2900 nM T22274 CH3SK8 58157594 IC50 = 177 nM T22274 CJ6MV1 58157631 IC50 = 162 nM T22274 CC5SH4 58157746 IC50 = 5 nM T22274 C4V7FY 58191950 IC50 > 32000 nM T22274 CPCA29 58191961 IC50 = 7.3 nM T22274 C7HF1L 58191965 IC50 > 32000 nM T22274 CR4BX0 58191982 IC50 > 32000 nM T22274 C8V1NK 58191988 IC50 > 32000 nM T22274 C8LWY9 58191997 IC50 > 32000 nM T22274 C3IQ9B 58191999 IC50 > 32000 nM T22274 CQB69R 58192003 IC50 > 32000 nM T22274 C5D4WO 58465584 IC50 = 2200 nM T22274 CK5W8N 58465588 IC50 = 110 nM T22274 C5K9LO 58465646 IC50 = 810 nM T22274 CP03LK 58465664 IC50 = 730 nM T22274 CX4IL2 58465681 IC50 = 32 nM T22274 CIG02Q 58465705 IC50 = 3500 nM T22274 CLD40J 58465708 IC50 = 33 nM T22274 C7S4IJ 58465719 IC50 = 150 nM T22274 C9LR0X 58465755 IC50 = 85 nM T22274 C5TON1 58465757 IC50 = 190 nM T22274 C3Q7IW 58465842 IC50 = 64 nM T22274 C4DN9F 58465859 IC50 = 280 nM T22274 C24SAM 58465863 IC50 = 130 nM T22274 C1MB4Q 59323957 IC50 > 30000 nM T22274 CK6LX0 59454220 IC50 > 30000 nM T22274 C2SDN1 59454252 IC50 > 30000 nM T22274 CO6A2S 59585196 IC50 = 150 nM T22274 CP2HK9 60148667 IC50 = 5600 nM T22274 C27DKW 60148711 IC50 = 1900 nM T22274 CS2E6C 60148712 IC50 = 5300 nM T22274 CPF50R 60148997 IC50 = 9700 nM T22274 CB7X2E 60151224 IC50 = 331 nM T22274 CY05OU 60151225 IC50 = 4630 nM T22274 CWO8H0 60152596 IC50 = 6950 nM T22274 CXW14A 60164619 IC50 = 31.62 nM T22274 C2A7CX 60164723 IC50 = 102 nM T22274 C7FI3C 60164834 IC50 = 125.89 nM T22274 C9A0HY 60164937 IC50 = 63.1 nM T22274 CQ8O3A 60168030 IC50 < 1 nM T22274 C45AHD 60198453 IC50 < 1 nM T22274 C61LTI 60198519 IC50 < 1 nM T22274 C0OL8Y 60198521 IC50 < 1 nM T22274 C5HEZ7 60198582 IC50 < 1 nM T22274 CKDC94 60198648 IC50 < 1 nM T22274 CQ1U0P 60200243 IC50 > 50000 nM T22274 C90PVD 63992786 IC50 = 695 nM T22274 CBN3L0 69950064 Ki = 2810 nM T22274 C6RFQ8 70676597 IC50 > 20000 nM T22274 CM4XB8 70681905 IC50 = 3390 nM T22274 CW5MP0 70681906 IC50 = 2690 nM T22274 CGYX13 70681907 IC50 = 1550 nM T22274 CPMZ01 70681908 IC50 = 1220 nM T22274 CM62BN 70682297 IC50 > 20000 nM T22274 C3PR4C 70684025 IC50 = 9550 nM T22274 C8R9XE 70684026 IC50 = 1070 nM T22274 CT64UC 70686159 IC50 = 450 nM T22274 C94YFZ 70686160 IC50 = 23180 nM T22274 CBZ8W0 70688300 IC50 = 13460 nM T22274 CS8PU0 70688301 IC50 = 24750 nM T22274 CBY8S3 70690302 IC50 = 58670 nM T22274 C0CQP5 70690303 IC50 = 8770 nM T22274 C8T1FV 70690304 IC50 = 1330 nM T22274 CQ1R3N 70692543 IC50 = 1100 nM T22274 C7VF1B 70692849 IC50 > 20000 nM T22274 C28UMB 70693708 IC50 = 2800 nM T22274 CGSM24 70694519 IC50 = 120 nM T22274 C49EGA 70694593 IC50 = 20200 nM T22274 CE67KO 70695508 IC50 > 100000 nM T22274 CX23AC 70696578 IC50 = 390 nM T22274 CW6F1J 70696579 IC50 = 13500 nM T22274 CQY1I6 70789579 Ki = 189 nM T22274 C2ED7S 71139195 IC50 = 2204 nM T22274 C4BWT1 71142064 IC50 = 2390 nM T22274 CQO45N 71142065 IC50 = 3628 nM T22274 C8JK7A 71142076 IC50 = 957 nM T22274 CS1K8D 71142081 IC50 = 454 nM T22274 C0ELR8 71142091 IC50 = 1100 nM T22274 CE4P1B 71142092 IC50 = 905 nM T22274 CV8B4P 71142094 IC50 = 637 nM T22274 CK6GL1 71142097 IC50 = 847 nM T22274 C2RI8V 71142100 IC50 = 306 nM T22274 C6L0JF 71142106 IC50 = 1023 nM T22274 C3D2KM 71142108 IC50 = 1006 nM T22274 CQU52J 71142109 IC50 = 661 nM T22274 C25CUJ 71142127 IC50 = 812 nM T22274 C96LSO 71142130 IC50 = 1085 nM T22274 C1KF3N 71142131 IC50 = 807 nM T22274 CQ2E6U 71142135 IC50 = 356 nM T22274 CW6GQ3 71449487 IC50 < 1 nM T22274 CCZ73P 71450111 IC50 = 139 nM T22274 CH2PV4 71450133 IC50 = 11.7 nM T22274 C37HBI 71451928 IC50 = 468 nM T22274 C4ZNG6 71451952 IC50 = 9.26 nM T22274 C0ES2V 71453199 IC50 = 1700 nM T22274 C3J9QZ 71453454 IC50 > 10000 nM T22274 C9NWA2 71453740 IC50 = 41.1 nM T22274 CQ1G6B 71453741 IC50 = 458 nM T22274 CEY13X 71453772 IC50 = 5.8 nM T22274 CXI80Y 71454842 IC50 < 1 nM T22274 C57ATO 71455172 IC50 > 10000 nM T22274 C6V4AT 71456615 IC50 < 1 nM T22274 C6B2HJ 71456958 IC50 > 10000 nM T22274 C57LCN 71457287 IC50 = 14 nM T22274 C76SGF 71457594 IC50 = 2400 nM T22274 C82RMX 71458474 IC50 < 1 nM T22274 C6C4OT 71458560 IC50 = 330 nM T22274 CM9A3I 71458827 IC50 > 10000 nM T22274 C2HZ7Q 71460412 IC50 = 6500 nM T22274 CEXJ68 71460922 IC50 = 60.3 nM T22274 CBK53U 71462097 IC50 = 2000 nM T22274 CXSN25 71462624 IC50 = 25.2 nM T22274 CES2C4 71462625 IC50 = 2.38 nM T22274 CQ7VL0 71467493 IC50 = 3710 nM T22274 C5BR1D 71467494 IC50 = 4320 nM T22274 C3PIK2 71467958 IC50 = 1100 nM T22274 CTNS49 71467959 IC50 = 1110 nM T22274 CQ6B2I 71467960 IC50 = 930 nM T22274 C0YXF2 71467961 IC50 = 1210 nM T22274 C1MH5Z 71467962 IC50 = 122.55 nM T22274 C7ESZ2 71467963 IC50 = 630 nM T22274 C45FCJ 71468055 IC50 = 2300 nM T22274 C3H0CR 71468158 IC50 = 180 nM T22274 CQ26IW 71468159 IC50 = 380 nM T22274 C6ZPJ4 71468160 IC50 = 9540 nM T22274 CJU64Z 71468161 IC50 = 61.49 nM T22274 CD8O7W 71468162 IC50 = 750 nM T22274 CSDO79 71468163 IC50 = 190 nM T22274 CN97RG 71468164 IC50 = 470 nM T22274 C5I0TX 71468273 IC50 = 500 nM T22274 CJKU04 71468274 IC50 = 5170 nM T22274 CZJ84E 71468275 IC50 = 4990 nM T22274 C6L0RV 71468277 IC50 = 1070 nM T22274 CAH65F 71468278 IC50 = 1750 nM T22274 CVP26X 71468393 IC50 = 950 nM T22274 CFW2I5 71468672 IC50 = 21.91 nM T22274 C01IKD 71468927 IC50 = 2240 nM T22274 CNXK19 71468928 IC50 = 1190 nM T22274 C0CX7P 71476624 Ki > 2500 nM T22274 C6QPH1 71476625 Ki > 2500 nM T22274 C3JLD4 71476626 Ki > 2500 nM T22274 C3OH6T 71476627 Ki > 2500 nM T22274 C7GY8U 71495390 IC50 = 26 nM T22274 CBE46I 71495482 IC50 = 15 nM T22274 CQ5FC3 71495575 IC50 = 20 nM T22274 CIQ3E7 71495576 IC50 = 27 nM T22274 CAL79Y 71495577 IC50 = 16 nM T22274 C1SXH7 71495578 IC50 = 5.6 nM T22274 C1Q8LP 71495673 IC50 = 69 nM T22274 CF72JS 71495674 IC50 = 217000 nM T22274 C3T7UP 71495675 IC50 = 53 nM T22274 CFQ2N9 71520536 IC50 = 51.7 nM T22274 C0LWJ6 71520631 IC50 = 26.9 nM T22274 CO28HI 71520716 IC50 = 18.1 nM T22274 CVA5Q7 71520717 IC50 = 55.7 nM T22274 C89SWX 71527724 IC50 = 280 nM T22274 C6S5JQ 71527847 IC50 = 376.7 nM T22274 C6KBD4 71534512 IC50 = 35 nM T22274 CT51EW 71534810 IC50 = 2 nM T22274 C7QN3O 71534812 IC50 = 1 nM T22274 C8M3HU 71537640 IC50 = 160 nM T22274 C2QML7 71537641 IC50 = 4 nM T22274 CZJX53 71537927 IC50 = 582 nM T22274 CU0ZE6 71537928 IC50 = 3 nM T22274 CH9FS7 71537929 IC50 = 15 nM T22274 CTW95A 71537931 IC50 = 1 nM T22274 CW3BT5 71537932 IC50 = 9380 nM T22274 C3C0RO 71538475 IC50 = 3 nM T22274 CIA28E 71538746 IC50 = 6 nM T22274 CFCV26 71538748 IC50 = 83 nM T22274 CY2T1Q 71538749 IC50 = 139 nM T22274 C4A6VJ 71538750 IC50 = 2 nM T22274 CG72NC 71538751 IC50 = 4 nM T22274 CDW81Y 71574856 IC50 = 1360 nM T22274 CX01BJ 71574948 IC50 = 8 nM T22274 CO8YU7 71574949 IC50 = 28 nM T22274 CX6I3N 71577043 IC50 = 1100 nM T22274 C7MW4N 71582992 IC50 = 125.89 nM T22274 CKR6U8 71583101 IC50 = 22 nM T22274 CBZ5S9 71583103 IC50 = 1.9 nM T22274 C3PSJ9 71583105 IC50 = 3.7 nM T22274 C21GHR 71624738 IC50 = 120 nM T22274 CBN92Q 71625222 IC50 = 85 nM T22274 CLW8K3 71625224 IC50 = 42 nM T22274 C53BQN 71625225 IC50 = 36 nM T22274 CCQ0U1 71625341 IC50 = 75 nM T22274 COZX76 71625342 IC50 = 260 nM T22274 CD09SV 71625344 IC50 = 81 nM T22274 CU65GH 71655059 IC50 = 139.7 nM T22274 CPS58L 71655136 IC50 = 51 nM T22274 CFW7Q9 71655137 IC50 = 69.5 nM T22274 C9S0UB 71655138 IC50 = 86.6 nM T22274 CU27EV 71655139 IC50 = 133.3 nM T22274 CO8R1Z 71655216 IC50 = 127.4 nM T22274 C0W6EK 71655283 IC50 = 34 nM T22274 C7HG0K 71655802 IC50 = 30 nM T22274 CV73YD 71660259 IC50 = 3430 nM T22274 CQ5UR0 71660260 IC50 = 8240 nM T22274 CQ5P0T 71660261 IC50 = 440 nM T22274 C8EIX0 71660262 IC50 = 760 nM T22274 CF2BS5 71660263 IC50 = 9830 nM T22274 CPJ4V7 71680913 IC50 = 36 nM T22274 C9X8KM 71680914 IC50 = 59 nM T22274 C4W2MA 71680915 IC50 = 34 nM T22274 C3KO9V 71680916 IC50 = 57 nM T22274 CN4X5O 71680917 IC50 = 2500 nM T22274 CWAM13 71680918 IC50 = 1300 nM T22274 CI9G3B 71681069 IC50 = 21 nM T22274 C5WZV9 71720123 IC50 = 372 nM T22274 CIR56T 71721558 IC50 > 100000 nM T22274 CCD18W 71721946 IC50 > 100000 nM T22274 CFUC24 71722010 IC50 = 9.6 nM T22274 CXMZ49 71732116 IC50 = 12 nM T22274 C0H9PY 71732117 IC50 = 43 nM T22274 CSI0W8 71732119 IC50 = 6 nM T22274 CWGF27 71732120 IC50 = 74 nM T22274 C0P8CH 71748076 IC50 = 9 nM T22274 CU4X2F 71761851 IC50 = 8 nM T22274 C7SK3L 71761852 IC50 = 8 nM T22274 CI2NH1 71761853 IC50 = 32 nM T22274 CORB04 71762088 IC50 = 13 nM T22274 CYG6O7 71762089 IC50 = 13 nM T22274 CUBP37 71765043 IC50 = 567 nM T22274 C1UA2B 71765044 IC50 = 221 nM T22274 C6U9VB 71769925 IC50 = 250 nM T22274 CIRH21 71769926 IC50 = 180 nM T22274 C26HDR 71769927 IC50 = 340 nM T22274 C5RXY7 71769928 IC50 = 230 nM T22274 CT1RZ2 71770054 IC50 = 1100 nM T22274 CTPJ18 71770057 IC50 = 430 nM T22274 C1TSQ4 71770058 IC50 = 1930 nM T22274 CVU1W6 71770059 IC50 = 3130 nM T22274 CHK58Q 71770060 IC50 = 790 nM T22274 CG3X4E 71770191 IC50 = 930 nM T22274 CJ87KH 71770193 IC50 = 550 nM T22274 C8J7IV 71770194 IC50 = 830 nM T22274 CN5D6Z 71770321 IC50 = 1140 nM T22274 C13MPI 71770439 IC50 = 480 nM T22274 C5K4ZC 71770562 IC50 = 4650 nM T22274 CTSK68 71811225 IC50 = 29 nM T22274 C1K6OW 71811226 IC50 = 24 nM T22274 CU3N9R 71811227 IC50 = 88 nM T22274 CS2L4B 71811228 IC50 = 15 nM T22274 CL4DT9 71811229 IC50 = 35 nM T22274 CK6DB4 71811230 IC50 = 33 nM T22274 CIM3G4 71811257 IC50 = 41 nM T22274 CHR8V0 71811259 IC50 = 11 nM T22274 CVL54T 71811261 IC50 = 79 nM T22274 CZR93K 71811262 IC50 = 43 nM T22274 C52NYO 71811289 IC50 = 13 nM T22274 CM8BE4 71811290 IC50 = 41 nM T22274 C0MV3O 71811291 IC50 = 1920 nM T22274 C7UYD4 71811292 IC50 = 32 nM T22274 C7XL3N 71811293 IC50 = 690 nM T22274 C4HBC5 71811294 IC50 = 14 nM T22274 CTA26S 71811295 IC50 = 8 nM T22274 CE89AK 71818242 IC50 > 20000 nM T22274 C8M3IX 71818243 IC50 > 20000 nM T22274 CKP5J7 71818244 IC50 > 20000 nM T22274 CT7L6G 72163687 Ki > 2500 nM T22274 CKE9D3 72163688 Ki > 2500 nM T22274 CI9H6L 72164895 IC50 = 2.7 nM T22274 CH68XV 72188554 IC50 = 7 nM T22274 CS5UL7 72195322 IC50 = 5218 nM T22274 CNC56Z 72204472 IC50 = 5900 nM T22274 CR59TH 72204473 IC50 > 100000 nM T22274 CB9L8Z 72204662 IC50 = 7720 nM T22274 CT7M6G 72204663 IC50 = 460 nM T22274 C1VG8U 72204664 IC50 = 1120 nM T22274 CC0XI1 72204665 IC50 = 9080 nM T22274 C4MW3U 72204666 IC50 > 100000 nM T22274 C98VDM 72204667 IC50 = 180 nM T22274 C4FKY5 72204850 IC50 > 100000 nM T22274 CU30CD 72205221 IC50 = 6500 nM T22274 C90FMR 72205411 IC50 = 400 nM T22274 CAC5Q7 72375561 IC50 = 50 nM T22274 C3WQV2 72375562 IC50 = 98 nM T22274 CC1W6J 72375670 IC50 = 1100 nM T22274 C1A4YW 72545684 IC50 = 8 nM T22274 CM3KS6 72696333 IC50 = 1060 nM T22274 CI2EH8 72696334 IC50 = 130 nM T22274 C0CM8Q 72696335 IC50 = 90 nM T22274 CG31RX 72696336 IC50 = 520 nM T22274 CJ3EH7 72696464 IC50 = 160 nM T22274 C1OA0T 72696465 IC50 = 40 nM T22274 C1I9TZ 72696466 IC50 = 214 nM T22274 CFU3V5 72696467 IC50 = 88 nM T22274 CTR52Z 72696598 IC50 = 405 nM T22274 C4O2ZT 72696599 IC50 = 42 nM T22274 C5N9BQ 72696600 IC50 = 357 nM T22274 CE87BF 72696601 IC50 = 84 nM T22274 CV09DJ 72734543 IC50 = 385.8 nM T22274 CS6LW0 72946640 IC50 = 5 nM T22274 CXM37Z 72946641 IC50 = 8 nM T22274 CQA16N 72946833 IC50 = 3 nM T22274 CNR7Z2 72946834 IC50 = 19 nM T22274 C12JYS 72946835 IC50 = 4 nM T22274 C5Y9XH 72946836 IC50 = 4 nM T22274 CVZR94 72946837 IC50 = 31 nM T22274 C8-AUG 72946838 IC50 = 8 nM T22274 CHQ39Y 72947043 IC50 = 3 nM T22274 CCST90 72947044 IC50 = 3 nM T22274 C7J3RH 72947045 IC50 = 4 nM T22274 CK10LZ 73292342 IC50 = 747 nM T22274 CPT58N 73333212 IC50 = 19 nM T22274 C0FC3H 73333213 IC50 = 52 nM T22274 CE8CB6 73333214 IC50 = 12000 nM T22274 CX3W1T 73333311 IC50 = 19 nM T22274 CC9VI3 73333312 IC50 = 79 nM T22274 CTBL47 73333313 IC50 = 76 nM T22274 C8C1OY 73333314 IC50 = 1300 nM T22274 C0FI1Z 73333416 IC50 = 120 nM T22274 C40IPG 73333417 IC50 = 2600 nM T22274 C21XQI 73345596 IC50 = 180 nM T22274 CDG47J 73346009 IC50 > 20000 nM T22274 C6H7IJ 73346010 IC50 > 20000 nM T22274 CD0WU2 73346011 IC50 > 20000 nM T22274 COBJ19 73347538 IC50 > 20000 nM T22274 C5FDJ0 73347611 IC50 > 10000 nM T22274 C92HFB 73349064 IC50 > 20000 nM T22274 C68LBO 73349131 IC50 < 0.2 nM T22274 CN24OK 73350652 IC50 = 7080 nM T22274 CAS8E2 73352138 IC50 > 20000 nM T22274 CB96UM 73352206 IC50 = 4060 nM T22274 CSP58Q 73353181 IC50 = 1440 nM T22274 CH6Z2L 73353182 IC50 = 5700 nM T22274 C0C2QO 73353595 IC50 > 20000 nM T22274 C59WMZ 73353596 IC50 > 20000 nM T22274 C1UDF8 73353597 IC50 > 20000 nM T22274 C0UQO1 73353605 IC50 = 2700 nM T22274 CUD02X 73355098 IC50 = 78 nM T22274 CXK86S 73355189 IC50 = 16 nM T22274 CGM2S4 73356727 IC50 > 10000 nM T22274 CNC6Q5 73505594 IC50 = 61 nM T22274 CPQ43R 73707550 IC50 = 0.5 nM T22274 CJ1DA8 73774764 IC50 = 164.4 nM T22274 CQ3K6G 73776326 IC50 = 142.2 nM T22274 CC4L0G 73776327 IC50 = 143.7 nM T22274 CZB6G7 73776472 IC50 = 308.2 nM T22274 CSRE84 73776614 IC50 = 101.7 nM T22274 C01FVX 73776616 IC50 = 185.6 nM T22274 C3UC9H 73891099 IC50 = 4600 nM T22274 C3YH9X 76314009 IC50 = 955 nM T22274 CL4JQ3 76331862 IC50 = 75 nM T22274 CTZ53J 76332759 IC50 = 780 nM T22274 C08CPW 76335428 IC50 = 6 nM T22274 C7JQU3 76335755 IC50 = 911 nM T22274 CKI74A 76853213 IC50 = 1200 nM T22274 CCR7L2 76853289 IC50 = 14000 nM T22274 C96LMJ 78323868 IC50 = 2.6 nM T22274 C5IAU4 78323870 IC50 = 3.8 nM T22274 CJ6Z0X 78324068 IC50 = 3600 nM T22274 C25ETN 78324161 IC50 = 1.8 nM T22274 C3U0KE 81689842 IC50 = 6200 nM T22274 CE1AN2 82017359 IC50 = 60000 nM T22274 CG5ZD9 86291495 IC50 = 58 nM T22274 C61VCD 86294741 IC50 = 4200 nM T22274 CBWV30 86294747 IC50 = 8800 nM T22274 CGF12C 86302517 IC50 = 150 nM T22274 C8O5PZ 86302518 IC50 = 550 nM T22274 CY5Q0E 86302520 IC50 = 6100 nM T22274 C06YBD 86302594 IC50 = 4.1 nM T22274 C3EM7H 86581004 IC50 = 430 nM T22274 C7UK3Y 86581005 IC50 = 92 nM T22274 CY64UM 86581152 IC50 = 630 nM T22274 CY5V7C 86581153 IC50 = 550 nM T22274 C1HE8I 86581432 IC50 = 290 nM T22274 CZM07I 86581434 IC50 = 110 nM T22274 C8ZQG9 86581435 IC50 = 440 nM T22274 C6M9PL 86765212 IC50 = 5.2 nM T22274 CIKP60 86765426 EC50 = 930 nM T22274 CPX2N3 86765427 EC50 = 1180 nM T22274 CS5I4Y 87261507 IC50 = 2 nM T22274 C8ZM2A 87400677 IC50 = 43 nM T22274 C5JIT0 87618609 IC50 > 32000 nM T22274 CRQO37 88005144 IC50 > 32000 nM T22274 CRAX13 88849486 IC50 = 510 nM T22274 CD3X6M 88849490 EC50 = 5900 nM T22274 CQ2LF5 88920533 IC50 = 6.17 nM T22274 C2U9LW 88981186 IC50 = 63.1 nM T22274 CBSM71 89514711 IC50 = 270 nM T22274 CR27YF 89827822 IC50 = 53 nM T22274 CD7J6C 90644927 IC50 = 180 nM T22274 C62GSL 90654859 IC50 = 293.6 nM T22274 CYW51P 90654946 IC50 = 408 nM T22274 CJH1S6 90654947 IC50 = 16700 nM T22274 CSR56C 90655296 IC50 = 12 nM T22274 C15WHB 90656724 IC50 = 280 nM T22274 CSDO81 90664458 Ki = 247 nM T22274 CI9M0E 90665809 IC50 = 930 nM T22274 C23GNF 90665810 IC50 = 1680 nM T22274 CY0P7X 90665811 IC50 = 1920 nM T22274 C0RX4B 90667452 IC50 = 420 nM T22274 C8HL5V 90667453 IC50 = 1740 nM T22274 C3IE7F 90667454 IC50 = 1290 nM T22274 C37GOB 90667455 IC50 = 980 nM T22274 C67UHD 91619090 IC50 = 112 nM T22274 C6JZT7 91619093 IC50 = 270 nM T22274 C5M9AK 91667421 IC50 = 2849 nM T22274 CJO6T1 91810840 IC50 = 25 nM T22274 CYJ12Q 91884636 IC50 = 3 nM T22274 C0FCU9 91938063 IC50 = 20.81 nM T22274 C34WIG 92045024 EC50 = 1600 nM T22274 CN5KS8 92135978 IC50 = 1300 nM T22274 CYO9J5 101879983 IC50 = 11.43 nM T22274 C9OC0F 101882265 EC50 = 3450 nM T22274 CDV40P 101882454 IC50 = 150 nM T22274 C0M1NK 101882456 IC50 = 230 nM T22274 CPUJ32 101882458 IC50 = 280 nM T22274 CVE07R 101882857 IC50 = 4610 nM T22274 C7Q6ID 101884982 IC50 = 1 nM T22274 CR46PQ 101884983 IC50 = 5 nM T22274 CRZ83C 101884989 IC50 = 21 nM T22274 C12GJX 102366363 IC50 = 30 nM T22274 CO25LD 102366364 IC50 = 1200 nM T22274 C8CER4 102366365 IC50 = 8900 nM T22274 CT7Z8F 102514716 IC50 = 199.3 nM T22274 CS2UL0 117829456 IC50 = 40 nM T22274 C7L4OT 117829461 IC50 = 130 nM T22274 C50VUN 117829462 IC50 = 86 nM T22274 CPW71E 117855070 IC50 = 1.7 nM T22274 CB68IV 117855071 IC50 = 1.6 nM T22274 CSU52M 118656852 IC50 = 9.4 nM T22274 CB6AJ9 118656853 IC50 = 8 nM T22274 CAF41G 118707835 IC50 = 60 nM T22274 C0P4EV 118707836 IC50 = 30 nM T22274 CC8KL3 118707837 IC50 = 4100 nM T22274 C9VI8U 118707838 IC50 > 20000 nM T22274 CRU9G3 118707839 IC50 > 20000 nM T22274 C9SWI4 118707840 IC50 > 20000 nM T22274 CW9UJ1 118707841 IC50 > 20000 nM T22274 CBYI69 118707842 IC50 = 16100 nM T22274 C45UYG 118709095 IC50 = 32000 nM T22274 C7QHE4 118712502 IC50 = 61 nM T22274 C8KSD6 118712503 IC50 = 135 nM T22274 C1JFZ7 118714371 IC50 = 64 nM T22274 CXF0U3 118714375 IC50 = 158 nM T22274 C2M5OR 118714376 IC50 = 65 nM T22274 CY4GN9 118714377 IC50 = 34 nM T22274 CRL92Y 118714414 IC50 = 1300 nM T22274 CR37MV 118714415 IC50 = 1600 nM T22274 C96XGO 118715268 EC50 = 690 nM T22274 C7P3KH 118715726 IC50 = 568.76 nM T22274 CK6UM0 118715727 IC50 = 23.99 nM T22274 CW85VZ 118715728 IC50 = 21.96 nM T22274 CYGT73 118715730 IC50 = 30 nM T22274 CCAM49 118715731 IC50 = 11.49 nM T22274 C37NXA 118715732 IC50 = 7.88 nM T22274 CEN1J3 118715733 IC50 = 5.58 nM T22274 CFD2B8 118715734 IC50 = 8.87 nM T22274 CO8TJ6 118715735 IC50 = 6.55 nM T22274 C90TIX 118715736 IC50 = 8.46 nM T22274 C14KQU 118715737 IC50 = 8.58 nM T22274 CMK8B7 118715738 IC50 = 26.99 nM T22274 CQ6V9M 118715739 IC50 = 12.04 nM T22274 CWM04T 118715740 IC50 = 19.68 nM T22274 CLYS39 118715741 IC50 = 5.37 nM T22274 C04XZU 118715742 IC50 = 16.87 nM T22274 CJ4FS3 118715743 IC50 = 43.16 nM T22274 C3BH1K 118715744 IC50 = 3.44 nM T22274 CA12OP 118715745 IC50 = 2.69 nM T22274 C51RTI 118715746 IC50 = 1.9 nM T22274 CFX16A 118715747 IC50 = 3.42 nM T22274 C5OWL1 118715748 IC50 = 9.28 nM T22274 C8AW9X 118715749 IC50 = 7.19 nM T22274 C2Y7ZC 118715750 IC50 = 15.1 nM T22274 CPB7C3 118719377 Ki = 2200 nM T22274 C09OGH 118719378 Ki = 3700 nM T22274 C32LCM 118719380 Ki = 3000 nM T22274 C8U6YR 118719381 Ki = 1900 nM T22274 C9Y0HV 118719382 Ki = 6000 nM T22274 CF8BR9 118719410 IC50 = 39 nM T22274 CCYU59 118719817 IC50 = 5 nM T22274 CSC47W 118720522 IC50 = 93.8 nM T22274 CUI51W 118720529 IC50 = 23.9 nM T22274 CCGH73 118720703 IC50 = 26900 nM T22274 CMV2W9 118721625 IC50 = 1 nM T22274 CF5TO3 118721859 IC50 = 5 nM T22274 CK97TZ 118721860 IC50 = 1 nM T22274 CYV30O 118721861 IC50 = 2 nM T22274 C5WYI1 118721862 IC50 = 1 nM T22274 CSMW25 118721863 IC50 = 87 nM T22274 C5B1KM 118721864 IC50 = 6 nM T22274 CG8LZ0 118721865 IC50 = 5300 nM T22274 CPCN23 118721866 IC50 = 1770 nM T22274 CM0A9U 118721867 IC50 = 2710 nM T22274 CN47HE 118733259 IC50 = 48800 nM T22274 CJLN15 118733260 IC50 = 5740 nM T22274 CQ9PB1 118733372 EC50 = 13500 nM T22274 CU8T7G 118733373 IC50 = 1070 nM T22274 C6OEU2 118733374 EC50 = 300 nM T22274 CW5JY8 118733375 EC50 = 1900 nM T22274 CI8G4X 118737400 IC50 = 10 nM T22274 C2F8TQ 118737455 IC50 = 7.4 nM T22274 C1T6WZ 118738004 IC50 > 10000 nM T22274 CZ61KV 118753026 IC50 = 62 nM T22274 CFI23Y 118753027 IC50 = 1100 nM T22274 C75LTK 118753189 IC50 = 4900 nM T22274 CM3FB8 118796366 IC50 = 3000 nM T22274 CFDT16 118868555 IC50 = 1.66 nM T22274 CZI72K 118868576 IC50 = 0.89 nM T22274 C8DVP1 118868599 Ki = 30.2 nM T22274 C9G4LD 118868621 Ki = 14.13 nM T22274 CC71KZ 118868652 IC50 = 2.38 nM T22274 CQT5I6 118868656 Ki = 6.51 nM T22274 CE3PD1 118868670 Ki > 20000 nM T22274 CTL06Q 118884494 IC50 = 4.54 nM T22274 C13ZMU 118884505 Ki = 0.08 nM T22274 C5L8QM 118884518 IC50 = 3.73 nM T22274 C67EYR 118884520 IC50 = 83.5 nM T22274 C52ZCO 118884581 IC50 = 9.32 nM T22274 CV0E3L 118884590 Ki = 0.51 nM T22274 CME8R7 118884591 Ki = 0.23 nM T22274 C4XJ7F 118884592 Ki = 4.15 nM T22274 CI54GX 118884613 Ki = 0.42 nM T22274 C49UIG 118884644 IC50 = 1.25 nM T22274 CB4FJ9 118884665 IC50 = 10.1 nM T22274 CP5TE9 118884676 Ki = 0.88 nM T22274 CVTL89 118884679 Ki = 0.16 nM T22274 CB84TO 121278998 IC50 = 20000 nM T22274 C9S5OK 121279020 IC50 > 50000 nM T22274 CVXA98 121304930 IC50 <= 500 nM T22274 CIA40K 121472983 IC50 = 37 nM T22274 CL3M2F 121499152 IC50 > 33330 nM T22274 C93JAV 122177622 IC50 = 23 nM T22274 C5HJ0C 122177623 IC50 > 10000 nM T22274 CSU97K 122177957 IC50 = 13 nM T22274 CRW9F3 122180812 IC50 = 1580 nM T22274 CJ42OQ 122180814 IC50 = 8340 nM T22274 CEW23B 122180816 IC50 = 189 nM T22274 C3TB4Y 122180820 IC50 = 4170 nM T22274 CC80JD 122180822 IC50 = 5010 nM T22274 CXPG14 122180823 IC50 = 71 nM T22274 CYCT17 122180828 IC50 = 1460 nM T22274 CP5ND8 122180830 IC50 = 648 nM T22274 CL16JS 122180834 IC50 = 8110 nM T22274 CE4AO3 122181046 IC50 = 230 nM T22274 C7XP2A 122181047 IC50 = 30 nM T22274 CYD03G 122181048 IC50 = 322 nM T22274 C0H9WU 122181882 IC50 = 35.16 nM T22274 C81QDF 122182040 IC50 = 126.48 nM T22274 C2VO8E 122184845 IC50 = 6.83 nM T22274 CGSF80 122184846 IC50 = 7.96 nM T22274 CN4H8Q 122184847 IC50 = 3.77 nM T22274 CT94PN 122184848 IC50 = 5.15 nM T22274 CI2X8M 122184849 IC50 = 40.88 nM T22274 C5HOK3 122184850 IC50 = 29.91 nM T22274 CZC3Q4 122184851 IC50 = 6.26 nM T22274 CQW6T3 122184852 IC50 = 10.95 nM T22274 CE4M7C 122184853 IC50 = 147.6 nM T22274 C7MT9U 122184854 IC50 = 29.5 nM T22274 C4AQ5H 122184855 IC50 = 25 nM T22274 C07UQJ 122184856 IC50 = 13.59 nM T22274 CST56N 122184857 IC50 = 32.06 nM T22274 C6K1HJ 122184858 IC50 = 38.7 nM T22274 CG19IO 122185146 IC50 = 54.25 nM T22274 CI4U2H 122185147 IC50 = 100 nM T22274 CU47DI 122185148 IC50 = 545.42 nM T22274 C9XMU5 122185149 IC50 = 351.85 nM T22274 C5QCF0 122185150 IC50 = 58.9 nM T22274 CSA1H8 122185151 IC50 = 286.26 nM T22274 CZG70W 122185152 IC50 = 304.02 nM T22274 CRTN32 122191260 IC50 = 1050 nM T22274 C28JVO 122192004 IC50 = 459 nM T22274 CF2D8U 122192005 IC50 > 10000 nM T22274 CV8YH0 122193364 IC50 = 18300 nM T22274 C1CI0Z 122193365 IC50 = 8900 nM T22274 C32LTK 122193367 IC50 = 8670 nM T22274 CE04LR 122193368 IC50 = 9890 nM T22274 CW1HK5 122195536 IC50 = 25.5 nM T22274 C5W8OZ 122376192 IC50 = 0.65 nM T22274 C2YLS8 122379529 IC50 = 55.61 nM T22274 CCI4M6 122379531 IC50 = 6.31 nM T22274 CZ74QC 122379532 IC50 = 12.14 nM T22274 CLZ19M 122379533 IC50 = 82.62 nM T22274 CL0X8K 122550124 IC50 > 1000 nM T22274 C24QLO 122550126 IC50 = 34 nM T22274 CNKM78 122550129 IC50 = 34 nM T22274 CL31AN 122550132 EC50 = 49.4 nM T22274 CJM9X5 122550134 IC50 = 49 nM T22274 CHS4F7 122550135 IC50 = 19 nM T22274 CB8J6A 122550165 IC50 > 1000 nM T22274 CZ6TC9 122550171 IC50 > 1000 nM T22274 CX87LD 122550174 IC50 = 111 nM T22274 C3V5ND 122550211 EC50 = 58.9 nM T22274 C64OME 122550212 IC50 = 196 nM T22274 C8PM6C 122550213 IC50 = 23 nM T22274 CAXY60 122550234 IC50 = 8.6 nM T22274 CAOH68 122550235 IC50 = 57 nM T22274 CR38WT 122550251 IC50 > 1000 nM T22274 CX61TL 122550293 IC50 > 1000 nM T22274 C63EYP 122601008 IC50 = 15 nM T22274 CCN03D 122601010 IC50 = 390 nM T22274 CZC01M 122601076 IC50 = 56 nM T22274 CXOB76 122619576 IC50 > 500 nM T22274 CSPQ08 122619751 IC50 > 500 nM T22274 CZE35C 122648343 IC50 = 7.78 nM T22274 C54RNT 122648367 IC50 = 6.4 nM T22274 C1UVI7 122648600 EC50 = 198.6 nM T22274 CMX59K 122648648 EC50 = 143.7 nM T22274 CVZ64I 122648649 IC50 = 2.7 nM T22274 CW03VD 126582837 IC50 = 58.35 nM T22274 C5UV6J 126582839 IC50 = 23.38 nM T22274 CR9AC4 126582841 IC50 = 89.35 nM T22274 C1HS3A 126582843 IC50 = 17.78 nM T22274 CFI58L 126582907 IC50 = 142.98 nM T22274 CMT02Y 126582908 IC50 > 10 nM T22274 C6W3RK 126648983 IC50 < 10 nM T22274 CLIW36 126649181 IC50 = 0.61 nM T22274 CTP62U 126649182 IC50 = 6 nM T22274 CM6YJ3 126649211 IC50 = 31 nM T22274 CJE89Y 126649237 IC50 < 10 nM T22274 CZ67DK 126738293 IC50 = 11.4 nM T22274 CEC14P 126738294 IC50 = 2.79 nM T22274 C59SEH 126738297 IC50 = 33.3 nM T22274 CLO14J 126738589 IC50 = 14.8 nM T22274 C3Q6FV 127024856 IC50 = 1100 nM T22274 CVFI87 127025051 IC50 = 2500 nM T22274 CQ39UE 127025078 IC50 = 313 nM T22274 C8FOZ4 127025172 IC50 = 5800 nM T22274 CE4CI8 127025178 IC50 = 26 nM T22274 CL8TF5 127025475 IC50 > 10000 nM T22274 C8VEY9 127025539 IC50 = 4900 nM T22274 CNSO40 127025540 IC50 = 880 nM T22274 CM38EU 127025541 IC50 = 10000 nM T22274 CY5T9P 127025646 IC50 = 27 nM T22274 CKJ6L8 127025647 IC50 = 97 nM T22274 CXVC21 127025656 IC50 = 81 nM T22274 CF4G7Q 127025769 IC50 > 10000 nM T22274 CIF74W 127025777 IC50 > 10000 nM T22274 CT2EK9 127025778 IC50 > 10000 nM T22274 CMWO84 127025780 IC50 > 10000 nM T22274 CWB73C 127025940 IC50 = 2770 nM T22274 C58JDE 127025947 IC50 = 1310 nM T22274 CQ32BA 127026381 IC50 = 7400 nM T22274 CQTF36 127026436 IC50 > 10000 nM T22274 C3Q8FL 127026437 IC50 > 10000 nM T22274 C2N1UD 127026438 IC50 > 10000 nM T22274 CWY63G 127026695 IC50 = 92 nM T22274 CO4JI5 127026735 IC50 = 40 nM T22274 CME4B7 127026736 IC50 = 210 nM T22274 CG34KC 127026737 IC50 = 90 nM T22274 CNX10Q 127026738 IC50 = 470 nM T22274 CJ0AI5 127026739 IC50 = 140 nM T22274 C60DIS 127026740 IC50 = 6900 nM T22274 C31UJC 127026741 IC50 > 10000 nM T22274 COI3S8 127026742 IC50 = 250 nM T22274 CCR4M7 127026743 IC50 = 330 nM T22274 CNH5P8 127026863 IC50 = 2540 nM T22274 C0BG8P 127027017 IC50 = 106 nM T22274 C1R4SF 127027021 IC50 = 241 nM T22274 CZR43H 127027067 IC50 = 450 nM T22274 CA1N7Y 127027068 IC50 = 1400 nM T22274 CE8CN3 127027069 IC50 = 850 nM T22274 CCG30L 127027070 IC50 = 220 nM T22274 CU84JL 127027071 IC50 = 4400 nM T22274 CSJ18X 127027150 IC50 = 182 nM T22274 CA58GI 127027171 IC50 = 59 nM T22274 CBT4S5 127027172 IC50 = 2180 nM T22274 C3UED2 127027173 IC50 = 110 nM T22274 CUSY71 127027174 IC50 = 195 nM T22274 C2OIE1 127027175 IC50 = 89 nM T22274 CT5VX3 127027322 IC50 > 10000 nM T22274 CJAE38 127027376 IC50 = 5000 nM T22274 C86OFN 127027393 IC50 = 5000 nM T22274 C8X6FT 127027394 IC50 > 10000 nM T22274 CK0J7H 127027395 IC50 > 10000 nM T22274 CTP3J4 127027396 IC50 > 10000 nM T22274 COU4I9 127027458 IC50 = 9370 nM T22274 CC0WJ2 127027462 IC50 = 311 nM T22274 CSZL73 127027477 IC50 = 1060 nM T22274 CY3P7V 127027483 IC50 = 500 nM T22274 C68TYH 127027490 IC50 = 1610 nM T22274 CA14VM 127027506 IC50 > 10000 nM T22274 CB9PL5 127027507 IC50 > 10000 nM T22274 CBOJ07 127027508 IC50 > 10000 nM T22274 CT18SH 127027509 IC50 > 10000 nM T22274 CJ8MQ3 127027677 IC50 = 30 nM T22274 CK53WF 127027678 IC50 = 167 nM T22274 C3EWH4 127027679 IC50 = 56 nM T22274 C1KWD3 127027680 IC50 = 84 nM T22274 CM3SZ5 127027716 IC50 = 1800 nM T22274 CM42UC 127027717 IC50 = 880 nM T22274 CBMZ67 127027718 IC50 = 2100 nM T22274 C1KVR2 127027719 IC50 > 10000 nM T22274 CD4T1B 127027794 IC50 = 3690 nM T22274 CG7Q3V 127027808 IC50 = 5070 nM T22274 C6JUF9 127027813 IC50 = 7660 nM T22274 CW8F7D 127027975 IC50 = 1300 nM T22274 C2QYV5 127027979 IC50 = 910 nM T22274 CX80AH 127027993 IC50 = 244 nM T22274 CO5E1V 127027994 IC50 = 235 nM T22274 CG8NU7 127027995 IC50 = 18 nM T22274 CZ7C3D 127028030 IC50 = 16.4 nM T22274 CLN54U 127028295 IC50 = 758 nM T22274 CL7EN6 127028391 IC50 = 89 nM T22274 CG91JU 127028631 IC50 = 2900 nM T22274 CW04XE 127028723 IC50 = 1910 nM T22274 CV07OM 127028943 IC50 = 22 nM T22274 C08RCM 127028973 IC50 = 27 nM T22274 C8FNI2 127029515 IC50 = 6500 nM T22274 CV9I8D 127030313 IC50 = 1000 nM T22274 CN6K5P 127030500 IC50 = 63 nM T22274 CCNK89 127030846 IC50 > 1000 nM T22274 CI8WG4 127031734 IC50 = 40 nM T22274 C40HQA 127031756 EC50 = 50.8 nM T22274 C9Q1WD 127031757 IC50 = 20 nM T22274 CC6FD8 127034721 IC50 = 1150 nM T22274 C4EH3T 127034722 IC50 > 50000 nM T22274 C2YXR7 127034902 IC50 > 50000 nM T22274 CD1TP7 127034929 IC50 = 248 nM T22274 CU1M3B 127034930 IC50 = 75.4 nM T22274 C4SI0Q 127034947 IC50 = 194 nM T22274 CMS1F6 127034948 IC50 = 77.2 nM T22274 C3VB0I 127034949 IC50 = 8.9 nM T22274 CQC2F9 127035098 IC50 = 17.5 nM T22274 CBP64A 127035107 IC50 = 3.76 nM T22274 CAXL98 127035256 IC50 > 10000 nM T22274 CBJG94 127035257 IC50 = 1730 nM T22274 C9ZF0D 127035369 IC50 = 43700 nM T22274 C29AJN 127035766 IC50 = 6.99 nM T22274 C4GI0F 127037614 IC50 = 69 nM T22274 C50FSZ 127038118 EC50 = 17700 nM T22274 C18FSM 127039340 IC50 = 34 nM T22274 CIO0G3 127039341 IC50 = 93 nM T22274 C12NJF 127039347 IC50 = 150 nM T22274 CZ8A1F 127041696 EC50 = 5000 nM T22274 C69IXG 127041845 IC50 = 360 nM T22274 CO72YC 127045674 IC50 = 90 nM T22274 CTG0U3 127045675 IC50 = 390 nM T22274 CD42EQ 127045676 IC50 = 400 nM T22274 C9K0TN 127045677 IC50 = 900 nM T22274 CK51QO 127045678 IC50 = 2300 nM T22274 CG13WB 127046056 IC50 = 8600 nM T22274 CIQA39 127046057 IC50 = 900 nM T22274 CC89WM 127046659 IC50 = 140 nM T22274 CR61BE 127046852 IC50 = 800 nM T22274 CXJM94 127046853 IC50 = 600 nM T22274 C42VYT 127046854 IC50 = 2900 nM T22274 CR6AH4 127046855 IC50 = 2400 nM T22274 CM76WI 127046917 IC50 = 150 nM T22274 CQ8LT6 127047324 IC50 = 90 nM T22274 CJ7YR6 127047335 IC50 = 130 nM T22274 CB0O4H 127047412 IC50 = 1000 nM T22274 C5OH2V 127047413 IC50 = 5100 nM T22274 CEUB27 127047550 IC50 = 1500 nM T22274 CU1M3Q 127047551 IC50 = 300 nM T22274 CKH4S0 127047552 IC50 = 150 nM T22274 C7TV8A 127047636 IC50 = 3100 nM T22274 C4N2BY 127047651 IC50 = 2500 nM T22274 C5SW8E 127047652 IC50 = 500 nM T22274 CE1K8N 127047653 IC50 = 120 nM T22274 C2KB3W 127048062 IC50 = 2600 nM T22274 CB8HR2 129104138 IC50 > 50000 nM T22274 CCH65A 129104183 IC50 = 12000 nM T22274 CFH8Q4 129104227 IC50 > 50000 nM T22274 C6HM5P 129104349 IC50 > 50000 nM T22274 CZTF90 129104374 IC50 > 50000 nM T22274 CUJ2P5 129104402 IC50 > 50000 nM T22274 CY3I6X 129104426 IC50 > 50000 nM T22274 C2UL9B 129626301 IC50 = 270000 nM T22274 CA9EV6 130205513 IC50 = 6900 nM T22274 C8KRX0 130205516 IC50 = 15000 nM T22274 CJ7CQ5 130205526 IC50 = 5000 nM T22274 CUHY85 130205779 IC50 = 3800 nM T22274 CGT6B0 130238385 Ki = 0.45 nM T22274 C1LHV5 130238407 IC50 = 13.6 nM T22274 CMWV13 130238420 Ki = 0.15 nM T22274 C2PQV1 130238444 IC50 = 3.78 nM T22274 CHRD59 130238461 IC50 = 8.03 nM T22274 C0GH4T 130238474 Ki = 0.32 nM T22274 C9ERM5 130238475 Ki = 72.24 nM T22274 C9DM7Y 130238477 IC50 = 24.1 nM T22274 CN64FB 130258064 IC50 = 3.26 nM T22274 C8IEV4 130258911 IC50 = 1.8 nM T22274 CUYQ28 130345472 IC50 = 2.3 nM T22274 C6OXE3 132134663 IC50 = 2.1 nM T22274 C8LZA2 132144667 IC50 = 2.83 nM T22274 CW65BE 132144806 IC50 = 3.35 nM T22274 CNQ89W 132144846 IC50 = 11.4 nM T22274 CG1FA7 132144994 IC50 = 403 nM T22274 C9Z0NG 132145156 IC50 = 9.48 nM T22274 C38PRW 132145237 IC50 = 7.4 nM T22274 C45LUW 132145558 IC50 = 525 nM T22274 C62VZX 132145722 IC50 = 4.78 nM T22274 C2OL5M 132145724 IC50 = 41.7 nM T22274 C6X3HG 132145728 IC50 = 0.795 nM T22274 C8O9DP 132157820 IC50 = 0.29 nM T22274 CGF1M3 132157829 IC50 = 4.24 nM T22274 COI43B 132157856 IC50 = 41.7 nM T22274 C01AYD 132157876 IC50 = 21.5 nM T22274 C70VDB 132157887 IC50 = 129 nM T22274 CM4TW3 132157914 IC50 = 2.33 nM T22274 C56AOB 132157932 IC50 = 1130 nM T22274 CX4L9R 132157933 IC50 = 25.3 nM T22274 CLUA95 132157961 IC50 = 5.89 nM T22274 CX18NK 132157991 IC50 = 3.25 nM T22274 CG3XB2 132157992 IC50 = 2.31 nM T22274 C0SK7Y 132158005 IC50 = 265 nM T22274 C0G9TV 132495274 IC50 = 3.2 nM T22274 COVK82 132515050 IC50 = 11 nM T22274 CJ25PE 132515051 IC50 = 3 nM T22274 C4L6UZ 132547258 IC50 = 50 nM T22274 CGBR54 132547259 IC50 = 66 nM T22274 CW4MP2 132547260 IC50 = 49 nM T22274 C1YO2Z 132547261 IC50 = 10 nM T22274 C1OJM4 132576507 IC50 = 10.18 nM T22274 CRQ0L4 132576509 IC50 = 16.72 nM T22274 C0Y2TP 132585192 IC50 = 281 nM T22274 CEK53Y 132600649 IC50 = 6 nM T22274 C4UAN3 134129876 IC50 = 83 nM T22274 C25EVA 134129883 IC50 = 22 nM T22274 CWRH43 134129994 IC50 = 92 nM T22274 CK2TM6 134130010 IC50 = 76 nM T22274 CYW6H1 134130165 IC50 = 183 nM T22274 C8CY7S 134131006 IC50 = 50 nM T22274 CQ7SN8 134131102 IC50 = 61 nM T22274 CYCS54 134131113 IC50 = 49 nM T22274 CQO23I 134131456 IC50 = 5 nM T22274 CHZ8A3 134131564 IC50 = 6830 nM T22274 CN9DL4 134132030 IC50 > 10000 nM T22274 CA7J2D 134132574 IC50 = 19.5 nM T22274 CDMJ75 134135414 IC50 = 13.6 nM T22274 CX93QK 134135812 IC50 = 1120 nM T22274 CA5P7T 134136358 IC50 = 36.7 nM T22274 CQ93RF 134136880 IC50 > 100000 nM T22274 CG21VI 134136955 IC50 = 45000 nM T22274 C53UTO 134137062 IC50 = 2 nM T22274 CYGZ85 134137500 IC50 = 13.8 nM T22274 CJC1E8 134137789 IC50 = 12.9 nM T22274 CI0DC7 134138196 IC50 = 2.5 nM T22274 C3RA6C 134138227 IC50 = 4.1 nM T22274 CSX58U 134139437 IC50 > 10000 nM T22274 C26PWD 134139689 IC50 = 2800 nM T22274 CK7EZ2 134139706 IC50 = 18.5 nM T22274 CCF0X1 134140501 IC50 = 9.5 nM T22274 C08YTI 134140697 IC50 = 5.89 nM T22274 C8CP1R 134141659 IC50 = 66 nM T22274 C75NRQ 134141877 IC50 = 2030 nM T22274 C62SVR 134142119 IC50 > 100000 nM T22274 CFJX74 134142865 IC50 = 395 nM T22274 CLI48U 134143743 IC50 = 47300 nM T22274 CUA26W 134143927 IC50 = 850 nM T22274 C7FXS5 134144592 IC50 = 2900 nM T22274 C9Y0KW 134144836 IC50 = 64000 nM T22274 CEDU72 134145690 IC50 = 15.8 nM T22274 C1E2ZW 134145921 IC50 = 510 nM T22274 CL9H5I 134146726 IC50 = 10000 nM T22274 CWRJ15 134147087 IC50 = 60000 nM T22274 C8K0XJ 134147090 IC50 > 10000 nM T22274 C8O9SN 134147898 IC50 = 28 nM T22274 CP14DK 134149339 IC50 = 14.3 nM T22274 CG9H5W 134150350 IC50 = 2600 nM T22274 CQ61SB 134150479 IC50 = 495 nM T22274 CM7H0R 134150543 IC50 = 94.2 nM T22274 CJX12K 134151832 IC50 = 107 nM T22274 CDX75O 134152551 IC50 = 170 nM T22274 CHJ2I6 134152624 IC50 > 100000 nM T22274 C2JV5X 134153768 IC50 > 100000 nM T22274 C96JCY 134153909 IC50 = 2.3 nM T22274 C2E8MV 134154228 IC50 = 15 nM T22274 CBY2R8 134156011 IC50 = 8.4 nM T22274 C8F1BP 134156083 IC50 = 899 nM T22274 C38DIF 134156853 IC50 = 600 nM T22274 CI4W7T 134156856 IC50 = 16 nM T22274 C4FLQ5 134157355 IC50 = 14000 nM T22274 CCN19D 134157542 IC50 = 53000 nM T22274 C1UP3S 134157845 IC50 = 36 nM T22274 C9DSR3 134159676 IC50 = 5100 nM T22274 C0X1HQ 134224487 IC50 > 40000 nM T22274 CZV43J 134283792 IC50 = 88 nM T22274 C62WXO 134283796 IC50 = 95 nM T22274 CO7K3N 134283799 IC50 = 160 nM T22274 CBQ17L 134283800 IC50 = 48 nM T22274 C1Y4TA 134283810 IC50 = 140 nM T22274 CV2YF7 134283813 IC50 = 140 nM T22274 C05FVT 134492522 IC50 > 10000 nM T22274 CWJ7D1 134611695 IC50 = 5 nM T22274 C1F6WZ 134812689 IC50 = 14 nM T22274 C7F0TV 134812690 IC50 = 60 nM T22274 CML7O0 134822021 IC50 = 53 nM T22274 C52IBY 134823859 IC50 = 270 nM T22274 C4Q6YP 135348847 IC50 = 1350 nM T22274 CU4F7J 135348851 IC50 = 200 nM T22274 CYJ61T 135348854 IC50 = 690 nM T22274 CJ1B8Z 135348856 IC50 = 190 nM T22274 C14FWK 135348858 IC50 = 12 nM T22274 CP90AW 135348876 IC50 = 4360 nM T22274 CJ9MO0 135348881 IC50 = 10 nM T22274 CR1Z8J 135348908 IC50 = 1990 nM T22274 CL89IZ 135357280 IC50 = 10 nM T22274 CVC58K 135357401 IC50 = 3 nM T22274 C1NE3V 135357406 IC50 = 7 nM T22274 CVE5F8 135357457 IC50 = 2 nM T22274 CHL50J 135357477 IC50 = 162 nM T22274 CL6QV8 135357481 IC50 = 368 nM T22274 C3B9KX 135357492 IC50 = 10 nM T22274 CN18BT 135357494 IC50 = 17 nM T22274 CIC92K 135357495 IC50 = 9 nM T22274 CD37GV 135357520 IC50 = 9 nM T22274 CE6I9K 135357548 IC50 = 6 nM T22274 C2HZ7W 135357575 IC50 = 52 nM T22274 C3I0YS 135357579 IC50 = 4 nM T22274 C5NM8Y 135357622 IC50 = 3 nM T22274 CT30QV 135357634 IC50 = 22 nM T22274 CRS4C5 135357638 IC50 = 1 nM T22274 CO41RI 135357654 IC50 = 7 nM T22274 CC49YE 135357669 IC50 = 8 nM T22274 C9I5UC 135357695 IC50 = 20 nM T22274 C78JCY 135357701 IC50 = 5 nM T22274 CDJ5N0 135357784 IC50 = 25 nM T22274 C58SLX 135357794 IC50 = 4 nM T22274 C5CA7O 135357811 IC50 = 5 nM T22274 CM91NE 135357815 IC50 = 12 nM T22274 C7JTQ8 135357826 IC50 = 56 nM T22274 CS0UK5 135357843 IC50 = 17 nM T22274 CFD84W 135357870 IC50 = 9 nM T22274 CTG57J 135357888 IC50 = 16 nM T22274 CCN71F 135358004 IC50 = 11 nM T22274 CAJ9L6 135358197 IC50 = 20 nM T22274 CG7P2I 135358203 IC50 = 9 nM T22274 CY73MD 135358206 IC50 = 6 nM T22274 CA3T8J 135358229 IC50 = 4 nM T22274 CR4N1V 135358300 IC50 = 26 nM T22274 C5D2MN 135358405 IC50 = 333 nM T22274 CS1V6A 135367138 IC50 > 50000 nM T22274 CVO59N 135367789 IC50 = 4700 nM T22274 CDY18W 135407493 IC50 = 24800 nM T22274 CW2I4R 135412048 IC50 > 100000 nM T22274 C7U0AV 135412194 IC50 = 13700 nM T22274 CI28ZH 135424818 IC50 = 709 nM T22274 CS54TL 135437514 IC50 = 12900 nM T22274 C36MUC 135441620 IC50 > 100000 nM T22274 CRB8M1 135444536 IC50 = 16700 nM T22274 CX5D6J 135446479 IC50 = 11200 nM T22274 C1TOK2 135449197 IC50 = 60900 nM T22274 CZ9GA7 135449434 IC50 = 230000 nM T22274 CW25GL 135462117 IC50 > 100000 nM T22274 CCL28F 135473106 IC50 > 100000 nM T22274 CYA60G 135497781 IC50 > 100000 nM T22274 C01EZF 135567459 IC50 = 2400 nM T22274 C8X5LO 135928012 Ki = 32 nM T22274 CI2YE8 135928628 IC50 = 40100 nM T22274 C50NIS 136025837 IC50 = 10800 nM T22274 C4OS0V 136025842 IC50 > 100000 nM T22274 CX7Z5B 136025843 IC50 > 100000 nM T22274 CB8EM9 136025984 IC50 > 100000 nM T22274 C49MUG 136025986 IC50 > 100000 nM T22274 C0OLS8 136030779 IC50 = 7900 nM T22274 CIA7R4 136030780 IC50 = 3200 nM T22274 C24LKN 136030781 IC50 = 1100 nM T22274 CH7Y3C 136086920 IC50 > 100000 nM T22274 C3VDL5 136086921 IC50 = 32600 nM T22274 C9GOB5 136086922 IC50 = 7200 nM T22274 CE3ZL7 136086923 IC50 > 100000 nM T22274 CJZ5F3 136086924 IC50 = 88000 nM T22274 CY9U0E 136173089 IC50 = 7 nM T22274 C32MPU 136173094 IC50 = 9 nM T22274 CXHY69 136230092 IC50 = 300 nM T22274 CWK9U7 136230093 IC50 = 310 nM T22274 CBS97C 136239447 IC50 > 20000 nM T22274 CE2F9G 136244081 IC50 > 20000 nM T22274 C9CH7S 136244085 IC50 > 20000 nM T22274 C5J2AX 136244086 IC50 > 20000 nM T22274 CILG36 136286746 IC50 = 268 nM T22274 C39WRP 136286747 IC50 = 2360 nM T22274 C7ZX5O 136286761 IC50 = 62 nM T22274 C9SV6G 136645392 IC50 = 1090 nM T22274 CANQ56 136645396 IC50 = 48 nM T22274 C9TGH1 136645397 IC50 = 217 nM T22274 C1F7JV 136645401 IC50 > 20000 nM T22274 C32LNQ 136645404 IC50 = 87 nM T22274 C4W0IE 136645405 IC50 = 340 nM T22274 CMIU28 136645406 IC50 = 10100 nM T22274 C3K2WL 136645410 IC50 = 33 nM T22274 CC1D0X 136645415 IC50 = 1600 nM T22274 C02RIK 136645417 IC50 = 4340 nM T22274 C8CT0Z 136645422 IC50 = 77 nM T22274 CAWT82 136645431 IC50 = 89 nM T22274 CBZ8Q1 136645433 IC50 = 12700 nM T22274 C21EJD 136645435 IC50 = 66 nM T22274 C1KTV3 136645436 IC50 = 1180 nM T22274 CK1B9W 136645438 IC50 = 42 nM T22274 C6QOP7 136645441 IC50 = 37 nM T22274 CMZ71T 136645444 IC50 = 815 nM T22274 CL47WS 136645445 IC50 = 192 nM T22274 C64BZR 136645447 IC50 = 10400 nM T22274 C7X1UL 136645449 IC50 = 110 nM T22274 CI9ZO7 136645454 IC50 = 256 nM T22274 CA3I8S 136645455 IC50 = 326 nM T22274 CRN16W 136645457 IC50 = 84 nM T22274 CGQ92L 136645458 IC50 = 89 nM T22274 CO5DN2 136645462 IC50 = 360 nM T22274 CRPN39 136645466 IC50 = 15 nM T22274 CL5X3G 136645467 IC50 = 168 nM T22274 C48HNY 136959539 IC50 = 1900 nM T22274 C1P8ZW 136959550 IC50 = 441 nM T22274 CKU95F 136966187 IC50 = 709 nM T22274 CFRG19 136985286 IC50 = 162 nM T22274 CE7F4O 136985287 IC50 = 584 nM T22274 CFPT21 136985288 IC50 = 87 nM T22274 CBH5Y0 136985291 IC50 = 1060 nM T22274 CDAK28 136985292 IC50 = 59 nM T22274 CQ9XW7 136985295 IC50 = 1790 nM T22274 C1M6NW 136985296 IC50 = 142 nM T22274 CJOA28 136985302 IC50 = 98 nM T22274 CP5NM4 137125260 IC50 > 100000 nM T22274 CANS59 137136982 IC50 > 20000 nM T22274 CDR9X0 137174935 IC50 = 33 nM T22274 CM1N3O 137226378 IC50 = 8850 nM T22274 C5AE3Q 137283418 IC50 > 20000 nM T22274 C5QIX1 137289788 IC50 = 130 nM T22274 C5X0YR 137289866 IC50 = 1250 nM T22274 CU70ZB 137289868 IC50 = 9640 nM T22274 CV6AN7 137289892 IC50 > 20000 nM T22274 CB14CI 137289900 IC50 = 5570 nM T22274 CLY69S 137289946 IC50 = 2350 nM T22274 CC5HA4 137290225 IC50 > 20000 nM T22274 C4RBC7 137290234 IC50 = 861 nM T22274 CKJ6Q4 137290238 IC50 = 2120 nM T22274 CR53GQ 137290273 IC50 = 91 nM T22274 C8DYG6 137290344 IC50 = 57 nM T22274 C9G3JB 137292402 IC50 = 379 nM T22274 C6MXL3 137292504 IC50 = 395 nM T22274 CAZ49O 137300702 IC50 = 79 nM T22274 CGE0J6 137300703 IC50 = 416 nM T22274 CDU43L 137300704 IC50 = 2330 nM T22274 CK0QG6 137300705 IC50 > 10000 nM T22274 C91IPL 137300706 IC50 = 5130 nM T22274 C5UYP8 137300707 IC50 > 20000 nM T22274 CHSG63 137300708 IC50 = 196 nM T22274 CX57MR 137300709 IC50 = 1920 nM T22274 C54KGS 137300710 IC50 = 373 nM T22274 CQD07Z 137300711 IC50 = 5370 nM T22274 C3I1CB 137300712 IC50 = 344 nM T22274 C2H0FQ 137314561 IC50 = 13 nM T22274 CR4S6Z 137314572 IC50 = 6 nM T22274 CI01YP 137314573 IC50 = 6 nM T22274 C0NE4B 137314592 IC50 = 5 nM T22274 CWM6Z2 137376574 Ki = 1.86 nM T22274 C3LUJ0 137487429 IC50 = 1030 nM T22274 C4VXT3 137553162 IC50 = 64 nM T22274 CA5OY1 137628667 IC50 = 70 nM T22274 C67EFJ 137628684 IC50 = 1.8 nM T22274 CX0PH5 137628685 IC50 = 190 nM T22274 CG23FD 137631444 IC50 > 30000 nM T22274 C9UQD2 137631509 IC50 > 30000 nM T22274 CP0JL9 137631552 IC50 > 30000 nM T22274 CP0BN3 137631704 Ki > 50000 nM T22274 C31MPL 137631726 IC50 = 2.8 nM T22274 CJ9GD5 137631769 IC50 > 30000 nM T22274 CQ54WK 137631915 IC50 > 30000 nM T22274 CD1L0I 137632135 IC50 > 30000 nM T22274 C1N8TU 137632249 Ki = 2.01 nM T22274 C6A4GK 137632422 IC50 > 30000 nM T22274 CQ4BK9 137632561 IC50 > 30000 nM T22274 CVB93K 137632723 IC50 = 2950 nM T22274 C9RWF1 137632979 IC50 > 30000 nM T22274 CI2G7B 137633049 IC50 > 30000 nM T22274 CMU42D 137633092 IC50 > 30000 nM T22274 CY08AM 137633123 IC50 > 30000 nM T22274 C84MIY 137633138 IC50 > 100000 nM T22274 CZY46A 137633389 IC50 = 4000 nM T22274 C1HL3I 137633415 IC50 > 30000 nM T22274 CS1LZ9 137633421 IC50 = 17.39 nM T22274 CM6V3G 137633491 IC50 = 35.79 nM T22274 C46IBX 137633497 IC50 = 12 nM T22274 CW8G1H 137633768 IC50 > 100000 nM T22274 C82QCH 137633786 IC50 = 108.48 nM T22274 CAUT87 137633927 IC50 = 110000 nM T22274 C5BZM4 137634010 IC50 = 5.28 nM T22274 C73PDL 137634086 IC50 > 100000 nM T22274 C1V8QE 137634156 IC50 = 21.7 nM T22274 C2OC5K 137634207 IC50 = 1.8 nM T22274 C8G4KJ 137634562 IC50 > 30000 nM T22274 CJ76DN 137634596 IC50 > 30000 nM T22274 C7JK8D 137634598 IC50 = 98.27 nM T22274 C7U1CE 137634604 IC50 > 30000 nM T22274 C28CEY 137634881 IC50 = 29.56 nM T22274 C90TSR 137634950 IC50 > 30000 nM T22274 CZ1FK2 137635119 IC50 > 50000 nM T22274 CHA4E3 137635225 IC50 = 1290 nM T22274 C6JVG9 137635398 IC50 = 1.4 nM T22274 CBMN61 137635405 IC50 > 30000 nM T22274 CAWZ25 137635575 IC50 = 6.8 nM T22274 CZ29MT 137635651 IC50 = 7160 nM T22274 C7N5BG 137635855 IC50 > 30000 nM T22274 C2KS3O 137635975 IC50 = 189 nM T22274 C2MB4U 137636234 IC50 = 1950 nM T22274 CA2S3J 137636481 IC50 = 2630 nM T22274 C63ZFX 137636534 IC50 = 148 nM T22274 C5GCO8 137636604 IC50 > 30000 nM T22274 CSY3E1 137636623 IC50 = 5000 nM T22274 C72SBN 137636632 IC50 > 30000 nM T22274 C9THE6 137636891 IC50 > 30000 nM T22274 CK1S0F 137637029 IC50 = 790 nM T22274 C8FH1S 137637247 IC50 = 2.9 nM T22274 CF3E8T 137637310 IC50 > 30000 nM T22274 C0VNM5 137637430 IC50 = 111.04 nM T22274 C5SZF4 137637483 IC50 = 25.3 nM T22274 C6MVX0 137637661 IC50 = 6430 nM T22274 C3H2GO 137637718 IC50 = 5370 nM T22274 CSH08B 137637787 IC50 = 4740 nM T22274 CEI0W2 137637915 IC50 = 410 nM T22274 CZU9E2 137637958 IC50 = 21.29 nM T22274 CMU93I 137637990 IC50 > 30000 nM T22274 C6X0AW 137638091 IC50 = 20.05 nM T22274 CMD89K 137638151 IC50 = 11580 nM T22274 CQ3DR6 137638257 IC50 = 5050 nM T22274 CO9UY1 137638342 IC50 > 30000 nM T22274 CW6F2I 137638447 IC50 = 35.94 nM T22274 C3RC2O 137638626 IC50 > 30000 nM T22274 CEMX30 137638687 IC50 > 30000 nM T22274 CTUL07 137638741 IC50 = 8.32 nM T22274 CTG6X0 137638748 IC50 > 30000 nM T22274 CX8Q4R 137638837 Ki = 0.48 nM T22274 CDWG31 137638917 IC50 > 100000 nM T22274 CZU31H 137638926 IC50 = 2870 nM T22274 CQ86FE 137638947 IC50 > 30000 nM T22274 C7IJC2 137639014 IC50 = 1700 nM T22274 C69IOZ 137639088 IC50 = 6.1 nM T22274 C0J8ZG 137639219 IC50 = 88 nM T22274 CUG0C9 137639328 IC50 > 10000 nM T22274 C2DIM1 137639536 IC50 = 1350 nM T22274 CJBF37 137639551 IC50 = 70.49 nM T22274 CW4DJ8 137639563 IC50 > 30000 nM T22274 CS9A6C 137639566 IC50 > 30000 nM T22274 CMI6Z0 137639764 IC50 = 2350 nM T22274 C3CD6L 137639796 IC50 = 791.6 nM T22274 COV42L 137639829 IC50 > 30000 nM T22274 CL02GC 137640047 IC50 = 4980 nM T22274 C06BYV 137640258 IC50 > 100000 nM T22274 C19GDO 137640291 IC50 = 87 nM T22274 CGKA54 137640295 IC50 > 30000 nM T22274 C7VIL6 137640304 IC50 = 5380 nM T22274 C0Q3ZW 137640468 IC50 = 19840 nM T22274 C7HF0W 137640828 IC50 = 4600 nM T22274 CS50ET 137641009 IC50 = 84.9 nM T22274 C39FQX 137641152 IC50 > 30000 nM T22274 CSA84O 137641263 IC50 = 3060 nM T22274 C3V4KQ 137641382 IC50 = 6 nM T22274 CI4PM3 137641395 IC50 > 30000 nM T22274 C4OEC3 137641520 IC50 = 320 nM T22274 C5JUR2 137641533 IC50 = 8.5 nM T22274 CS1K3I 137641616 IC50 > 30000 nM T22274 C38HXT 137641735 IC50 = 6350 nM T22274 CV19SL 137642038 IC50 > 30000 nM T22274 C7HKW1 137642159 IC50 = 41.43 nM T22274 CAF1N9 137642211 IC50 = 42.52 nM T22274 C40JZA 137642448 IC50 > 30000 nM T22274 CKPB85 137642609 IC50 = 0.9 nM T22274 CY02GK 137642671 IC50 > 30000 nM T22274 C7MOD4 137642692 IC50 = 39.93 nM T22274 CXV15S 137642770 IC50 = 604 nM T22274 C1PRH5 137642860 IC50 = 135 nM T22274 C37BJQ 137642900 IC50 > 100000 nM T22274 CQF49N 137643043 IC50 = 14400 nM T22274 CF42GI 137643288 IC50 = 36.61 nM T22274 C5QC2N 137643440 IC50 = 24.8 nM T22274 C4V1WC 137643841 IC50 = 990 nM T22274 CB59SN 137643993 IC50 = 58.54 nM T22274 CC38FN 137644424 IC50 > 30000 nM T22274 CVQ4J0 137644605 IC50 > 30000 nM T22274 CX37VS 137644658 IC50 > 30000 nM T22274 CPL3J1 137645258 IC50 > 30000 nM T22274 C8GNS5 137645287 IC50 = 275.35 nM T22274 C8XAR3 137645372 IC50 > 30000 nM T22274 C8WPM4 137645400 IC50 = 41.8 nM T22274 CI8YV3 137645454 IC50 = 7500 nM T22274 C05LHW 137645511 IC50 > 30000 nM T22274 CX3E0H 137645675 IC50 > 100000 nM T22274 CYSU67 137645967 IC50 > 30000 nM T22274 C8HKU4 137646033 IC50 = 87.6 nM T22274 CT98PM 137646118 IC50 = 170 nM T22274 CV7F6C 137646133 IC50 = 580 nM T22274 CMJ7D9 137646202 IC50 > 30000 nM T22274 CN08DL 137646214 IC50 > 30000 nM T22274 CNT3Y7 137647005 IC50 = 119.94 nM T22274 C4I9YE 137647260 IC50 = 6920 nM T22274 CX8C9V 137647325 IC50 > 30000 nM T22274 CA0V2Q 137647353 IC50 = 106 nM T22274 CHW8X4 137647384 IC50 > 30000 nM T22274 CGMN16 137647616 Ki > 50000 nM T22274 CM65KH 137647813 IC50 = 14.4 nM T22274 C5AFM1 137647889 IC50 = 56.02 nM T22274 CG4ZT1 137647906 IC50 = 19.6 nM T22274 CZ2RN9 137647935 IC50 > 30000 nM T22274 C5IK9F 137648357 IC50 = 71.38 nM T22274 C0K5AL 137648444 IC50 = 550 nM T22274 C8S2TO 137648573 IC50 = 6270 nM T22274 C0VAB8 137648585 IC50 > 30000 nM T22274 CPK7Y5 137648623 IC50 = 8460 nM T22274 CL0XW1 137648762 IC50 = 1890 nM T22274 CR0P6Z 137648837 IC50 = 2050 nM T22274 CG2PL8 137648996 IC50 = 1760 nM T22274 C05DNH 137649390 IC50 > 30000 nM T22274 CO20AE 137649565 IC50 > 30000 nM T22274 C7MHG2 137649586 IC50 = 7.1 nM T22274 CGK2M9 137649620 IC50 = 2800 nM T22274 CM15FY 137649624 IC50 = 201 nM T22274 CDXE54 137649646 Ki > 50000 nM T22274 CE67ZS 137649860 IC50 = 241 nM T22274 CH0ES8 137650022 IC50 > 30000 nM T22274 CRP0D7 137650200 IC50 = 11.87 nM T22274 C4MC5X 137650991 IC50 > 30000 nM T22274 C3VM4T 137651193 IC50 = 4.68 nM T22274 CK6X4L 137651315 IC50 = 140000 nM T22274 C4GNA5 137651338 IC50 > 30000 nM T22274 CEP9R0 137651700 IC50 = 16.7 nM T22274 CA4FM3 137651729 IC50 = 49.5 nM T22274 CH38FU 137651757 IC50 = 180000 nM T22274 C8PWX1 137651771 IC50 > 30000 nM T22274 CGE1Z5 137651786 IC50 = 16000 nM T22274 CD89ZR 137651966 IC50 > 30000 nM T22274 C3EQ0D 137651991 IC50 = 16.87 nM T22274 CT05IE 137651994 IC50 = 2330 nM T22274 CFLX25 137652000 IC50 = 96.4 nM T22274 CH0TI5 137652048 IC50 = 129.4 nM T22274 CH3B5G 137652131 IC50 > 30000 nM T22274 C8NHK9 137652359 IC50 > 100000 nM T22274 C5FHD3 137652442 IC50 = 0.8 nM T22274 CB15PI 137652670 Ki > 50000 nM T22274 C83RBI 137652888 IC50 = 1740 nM T22274 CPI06O 137652951 IC50 = 36.98 nM T22274 C3QX5N 137653295 IC50 > 100000 nM T22274 C61VOF 137653427 IC50 = 1980 nM T22274 COG3A4 137653572 IC50 = 65.1 nM T22274 CXZ5J3 137654094 IC50 = 214 nM T22274 C1OAE9 137654162 IC50 = 12120 nM T22274 CIW9C6 137654210 Ki = 0.7 nM T22274 C3FEM8 137654512 IC50 = 89.3 nM T22274 C39QLZ 137654517 IC50 = 36.5 nM T22274 C1HE8S 137654622 IC50 = 8.21 nM T22274 CFQ4T2 137654668 IC50 > 30000 nM T22274 CCR5B3 137654793 IC50 = 1 nM T22274 C0I1UW 137654820 IC50 = 534 nM T22274 C1SBN5 137654946 IC50 = 64.5 nM T22274 CLWF87 137655165 IC50 > 30000 nM T22274 CS50BH 137655597 IC50 > 30000 nM T22274 CN70IL 137655615 IC50 = 34 nM T22274 CZ5Y4F 137655761 IC50 = 16 nM T22274 C5EB0H 137655853 IC50 = 8.35 nM T22274 C71ZNJ 137656226 IC50 = 8.01 nM T22274 CIA0V1 137656228 IC50 > 30000 nM T22274 CI6R3W 137656303 Ki > 50000 nM T22274 C0NR1V 137656498 IC50 = 10.8 nM T22274 CRP0T2 137656638 IC50 = 63 nM T22274 C76OGQ 137656942 IC50 = 8 nM T22274 CY8A2I 137656945 IC50 = 392.7 nM T22274 C5BM7T 137657586 IC50 > 100000 nM T22274 CR6B5H 137657803 IC50 = 5100 nM T22274 C21XDS 137657845 IC50 = 270 nM T22274 C1DL3P 137657892 Ki > 50000 nM T22274 CYLD90 137658075 IC50 = 10.72 nM T22274 CN0C1E 137658519 IC50 > 30000 nM T22274 C8D2GT 137658785 Ki > 50000 nM T22274 COC9D2 137658833 IC50 > 30000 nM T22274 C8BZM7 137658924 IC50 = 3.56 nM T22274 C9D7NR 137659196 IC50 > 100000 nM T22274 C8FQ2G 137659331 Ki = 1.78 nM T22274 C6XWP9 137659968 IC50 = 138.13 nM T22274 CM0OE5 137660128 IC50 = 43.1 nM T22274 CW5FQ4 137660152 IC50 = 1570 nM T22274 CLWU57 137660171 IC50 > 100000 nM T22274 C7JGX8 137660397 IC50 = 33.84 nM T22274 C3Q7PX 137660404 IC50 = 3750 nM T22274 C02BSL 137661253 IC50 = 19.17 nM T22274 C5VR2U 137661620 IC50 = 0.14 nM T22274 C2RNY3 137661648 IC50 = 2610 nM T22274 C4B9EG 137661742 IC50 = 63.9 nM T22274 CO7Q1H 137661848 IC50 = 8900 nM T22274 CEJI95 137661885 IC50 = 600 nM T22274 CEF18M 137661927 IC50 > 100000 nM T22274 CQAY45 137662133 IC50 = 16170 nM T22274 CA51OM 137662221 IC50 = 27 nM T22274 CYZ43W 137662281 IC50 = 20.9 nM T22274 CM3UF7 137700779 IC50 > 10000 nM T22274 CAQ62X 137701235 Ki = 130 nM T22274 CXV84M 138377596 IC50 = 14 nM T22274 CVA12U 138377601 Ki = 1.6 nM T22274 C7EM3I 138393071 IC50 = 3.92 nM T22274 C4NFS3 138393072 IC50 = 17.5 nM T22274 CA3C4O 138454792 IC50 = 6.6 nM T22274 CIT72O 139302883 IC50 = 2.38 nM T22274 CN1TH8 139302889 IC50 = 41.65 nM T22274 C0R1MD 139302991 IC50 = 14.02 nM T22274 C3GJQ8 139303021 IC50 = 18.51 nM T22274 CN73DV 139303049 IC50 = 211 nM T22274 CFAU90 139303050 IC50 = 14.15 nM T22274 CKQB30 139303051 IC50 = 19.08 nM T22274 CN2UH1 139303146 IC50 = 1.59 nM T22274 CE81VG 139303149 IC50 = 2.02 nM T22274 C9DJ3B 139303559 IC50 = 18.31 nM T22274 C78AJB 140747740 IC50 = 100 nM T22274 C4KL9C 140747745 IC50 <= 100 nM T22274 C60FTR 140747751 IC50 <= 100 nM T22274 C13JZX 141522811 IC50 = 2600 nM T22274 CHS9N0 141728829 IC50 = 13 nM T22274 C9H8PX 141728841 IC50 = 41 nM T22274 CBV2K5 141728842 IC50 = 29 nM T22274 C2HF9A 141728845 IC50 = 300 nM T22274 C4RGY1 141728867 IC50 = 310 nM T22274 CH9K7L 141733188 IC50 = 22 nM T22274 C7XI0V 141764754 IC50 = 56 nM T22274 C3DCP2 142446438 IC50 = 24 nM T22274 CXC85I 142452063 IC50 = 3 nM T22274 C1OG5Z 142452080 IC50 = 136 nM T22274 C0ODS9 142452243 IC50 = 25 nM T22274 CX0E9B 142505968 IC50 = 39 nM T22274 C9G5ZW 142505990 IC50 = 889 nM T22274 CBJC50 142505992 IC50 = 2169 nM T22274 CJ5GT3 142506013 IC50 = 362 nM T22274 C7N8LV 142506025 IC50 = 37 nM T22274 CKBF56 142506033 IC50 = 36 nM T22274 CU03GW 142506036 IC50 = 8 nM T22274 C74MXW 142506065 IC50 = 69 nM T22274 C1PNM8 142506077 IC50 = 22 nM T22274 CX6BQ7 142506102 IC50 = 77 nM T22274 CY3BM0 142506119 IC50 = 45 nM T22274 CFJ6X3 142506136 IC50 = 4 nM T22274 CL3N4D 142506147 IC50 = 4 nM T22274 CC6MD0 142506155 IC50 = 1238 nM T22274 C05QOM 142506157 IC50 = 2699 nM T22274 CQI7B8 142506163 IC50 = 169 nM T22274 CLND62 142506170 IC50 = 431 nM T22274 CGNQ74 142506189 IC50 = 5 nM T22274 CT3U9R 142506192 IC50 = 28 nM T22274 CP71ZJ 142506208 IC50 = 3 nM T22274 C1T3IQ 142506210 IC50 = 5 nM T22274 CEGV67 142506220 IC50 = 10 nM T22274 CP5HF8 142506225 IC50 = 6 nM T22274 C1U3CA 142506238 IC50 = 4 nM T22274 C8GVK9 142506253 IC50 = 14 nM T22274 CW5BY1 145865295 IC50 = 17 nM T22274 CGU3V9 145865296 IC50 = 149 nM T22274 C0F2JV 145865297 IC50 = 314 nM T22274 C1COW3 145948735 IC50 = 181 nM T22274 CZ6D7U 145948737 IC50 = 2030 nM T22274 CL1T5W 145948741 IC50 = 361 nM T22274 C1GMF5 145948743 IC50 = 2.85 nM T22274 CCEB28 145948752 IC50 = 120 nM T22274 CTO5X4 145948791 IC50 = 32.9 nM T22274 CP98HY 145948798 IC50 = 106 nM T22274 C43XJI 145948810 IC50 = 620 nM T22274 C3JMP9 145948813 IC50 = 70.9 nM T22274 C7K1WB 145948814 IC50 = 31.4 nM T22274 CFU6J8 145948816 IC50 = 5350 nM T22274 CG1Y3W 145948818 IC50 = 43.8 nM T22274 CAY43C 145948836 IC50 > 10000 nM T22274 CKI3Y2 145948841 IC50 = 7.29 nM T22274 C7JWF3 145948843 IC50 = 41 nM T22274 CJG3B6 145948850 IC50 = 5.89 nM T22274 CGKI09 145948851 IC50 = 178 nM T22274 CZ16SK 145948852 IC50 = 31.9 nM T22274 CA6W8I 145948853 IC50 = 919 nM T22274 CF0Q3C 145948854 IC50 = 1230 nM T22274 CTEI37 145948871 IC50 = 3.61 nM T22274 C0VTX8 145948874 IC50 > 10000 nM T22274 C8FHP2 145948903 IC50 = 145 nM T22274 C7RLZ8 145948904 IC50 = 2170 nM T22274 CE4WS8 145948905 IC50 = 4.72 nM T22274 C1KO6S 145948906 IC50 = 269 nM T22274 C5EKH9 145948907 IC50 = 10.3 nM T22274 C5HL4D 145948914 IC50 = 95.3 nM T22274 C74UFN 145948956 IC50 = 18.9 nM T22274 CY09KL 145948957 IC50 = 14.7 nM T22274 CH91ER 145948958 IC50 = 24.5 nM T22274 CE38KZ 145948959 IC50 = 14.3 nM T22274 CE15JW 145948961 IC50 = 30.9 nM T22274 CN6YM2 145948964 IC50 = 3560 nM T22274 CY49SE 145948983 IC50 = 5660 nM T22274 CH0UZ1 145948985 IC50 > 10000 nM T22274 C7Y5PK 145948986 IC50 = 31.3 nM T22274 CY1KB9 145949010 IC50 = 6.67 nM T22274 C1EF9X 145950102 IC50 = 261 nM T22274 CRKM19 145950884 IC50 = 0.64 nM T22274 CV3QO5 145951170 IC50 = 8.5 nM T22274 CRSM78 145952088 IC50 > 160000 nM T22274 CFE4G6 145952135 IC50 = 290 nM T22274 CKG98W 145953085 IC50 = 139 nM T22274 C7I0VX 145953295 IC50 = 1025 nM T22274 C5EKX3 145954597 IC50 = 14 nM T22274 CM53ZB 145954785 IC50 = 50 nM T22274 CGP9X1 145955496 IC50 = 276 nM T22274 CFG58P 145957238 IC50 = 1790 nM T22274 CGC4T2 145958633 IC50 = 200 nM T22274 C3L8IE 145958641 IC50 = 419 nM T22274 CO05IK 145959360 IC50 = 74 nM T22274 C9IV1C 145959866 IC50 = 5.9 nM T22274 CE3T9X 145960682 IC50 = 2 nM T22274 CCKW65 145960815 IC50 < 10 nM T22274 CK1XI0 145960971 IC50 > 10000 nM T22274 C5OI0Y 145961494 IC50 > 10000 nM T22274 CB9G4Q 145961803 IC50 = 4 nM T22274 C12XQF 145961873 IC50 = 82 nM T22274 CRZ1M3 145962635 IC50 = 2800 nM T22274 C1X5EO 145962694 IC50 = 6.2 nM T22274 CXZ12B 145962724 IC50 < 10 nM T22274 CDR1E6 145962762 IC50 > 10000 nM T22274 C3PWD4 145964064 IC50 = 108 nM T22274 C2FI9K 145964537 IC50 = 218 nM T22274 CF95MI 145964579 IC50 = 33 nM T22274 CDY56B 145964885 IC50 = 751 nM T22274 C5CIX3 145965000 IC50 = 250 nM T22274 CB51JU 145965019 IC50 = 24500 nM T22274 CWX1T4 145965266 IC50 = 38 nM T22274 CK18TW 145966262 IC50 = 147 nM T22274 C9XLE7 145966296 IC50 = 27700 nM T22274 CJAE67 145966594 IC50 = 11.9 nM T22274 CTUF34 145966712 IC50 = 72 nM T22274 C56LKF 145966734 IC50 = 64 nM T22274 C0SG7F 145966799 IC50 = 78 nM T22274 CTRI57 145966861 IC50 = 6700 nM T22274 C1TSI7 145966890 IC50 = 242 nM T22274 C19POY 145967140 IC50 = 16.4 nM T22274 CV0TU5 145967196 IC50 = 69 nM T22274 C93JKN 145967593 IC50 = 20 nM T22274 CD82XB 145967610 IC50 = 36 nM T22274 C7OG1D 145967698 IC50 = 540 nM T22274 C5RPQ9 145967832 IC50 = 16 nM T22274 CI1ZD2 145967851 IC50 = 167 nM T22274 CR59HK 145967905 IC50 = 275 nM T22274 C95SNQ 145967968 IC50 = 359 nM T22274 CX0OD9 145968046 IC50 = 51.6 nM T22274 CES7W6 145968087 IC50 = 69 nM T22274 CSO4I7 145968364 IC50 > 5000 nM T22274 C2XS8E 145968675 IC50 = 168 nM T22274 CSJ81Y 145968726 IC50 = 1420 nM T22274 CG0S9U 145968824 IC50 = 326 nM T22274 CIA79M 145968985 IC50 = 8 nM T22274 C27YHM 145969456 IC50 = 22 nM T22274 CV53YN 145969651 IC50 = 35 nM T22274 C0K6XS 145969789 IC50 = 29 nM T22274 CUI37A 145969799 IC50 = 126.9 nM T22274 CWU27Z 145969804 IC50 = 8 nM T22274 CZ80EP 145969996 IC50 = 27 nM T22274 CFL68X 145970091 IC50 = 40500 nM T22274 C7TSV2 145970161 IC50 = 1057 nM T22274 CG5OK8 145970171 IC50 = 29 nM T22274 C3FQ0V 145970292 IC50 = 1800 nM T22274 CBR60K 145970453 IC50 = 107 nM T22274 C0E2UO 145970598 IC50 = 1 nM T22274 CI43DY 145970786 IC50 = 562 nM T22274 C63KEL 145970838 IC50 = 6300 nM T22274 C7UG3O 145971121 IC50 = 2820 nM T22274 C7VD9I 145971506 IC50 = 0.87 nM T22274 C7K1AJ 145971681 IC50 = 46 nM T22274 C8QM6W 145972270 IC50 = 1540 nM T22274 CS79UB 145972882 IC50 = 59 nM T22274 C76MET 145972988 IC50 = 132 nM T22274 CW0T7A 145973234 IC50 = 143 nM T22274 CO51JK 145973368 IC50 = 2.7 nM T22274 C4HTO2 145973543 IC50 = 1180 nM T22274 CSR50O 145973656 IC50 = 5900 nM T22274 C71FKO 145973698 IC50 = 385 nM T22274 CVM0Z3 145974125 IC50 = 848 nM T22274 C8A3YR 145974135 IC50 = 65 nM T22274 CYS37Z 145974282 IC50 = 41 nM T22274 C8YEJ9 145974425 IC50 = 9.25 nM T22274 C0PI8K 145974714 IC50 = 281 nM T22274 CZL05M 145975187 IC50 = 14100 nM T22274 CE8I5V 145975869 IC50 = 1810 nM T22274 CU65BZ 145976000 IC50 = 34000 nM T22274 C7ANI4 145976192 IC50 = 290 nM T22274 CMUA94 145976675 IC50 = 2750 nM T22274 CN6UO4 145977003 IC50 = 972 nM T22274 CKAQ67 145977127 IC50 = 15.5 nM T22274 CT5JQ9 145977224 IC50 = 157 nM T22274 CVNW49 145977244 IC50 = 345 nM T22274 C7J4SO 145977290 IC50 = 98 nM T22274 CS7K9I 145977545 IC50 = 293 nM T22274 CNTC23 145977597 IC50 = 40 nM T22274 CLY4Z5 145977632 IC50 = 620 nM T22274 CP53JS 145977717 IC50 = 7.1 nM T22274 C2WF3K 145978074 IC50 = 103 nM T22274 CLB32U 145978082 IC50 = 58 nM T22274 CDS2R6 145978162 IC50 = 178 nM T22274 C54RKV 145978707 IC50 = 34 nM T22274 COR40V 145978805 IC50 = 6.73 nM T22274 C7X4LZ 145978932 IC50 > 40000 nM T22274 C7TAL5 145979161 IC50 = 1.44 nM T22274 C9BJW3 145979532 IC50 = 19 nM T22274 CCV92M 145979587 IC50 = 35 nM T22274 CFT50A 145979673 IC50 = 2.4 nM T22274 CZ7IQ9 145979841 IC50 = 0.93 nM T22274 CZMP56 145980566 IC50 = 1780 nM T22274 CIM41N 145980574 IC50 = 1490 nM T22274 CDC6Y5 145980590 IC50 = 188 nM T22274 CWH40Y 145980630 IC50 = 3.7 nM T22274 CX94BD 145980658 IC50 = 0.81 nM T22274 C09BPI 145980773 IC50 = 3.5 nM T22274 CI1QV5 145980850 IC50 = 178 nM T22274 C2HA8W 145981067 IC50 = 60.7 nM T22274 C9ZT8Y 145981096 IC50 = 117 nM T22274 C1ZI9A 145981290 IC50 = 863 nM T22274 COG0N1 145981347 IC50 = 3150 nM T22274 CBZ2A7 145981846 IC50 = 181 nM T22274 CFR1P8 145981954 IC50 = 31 nM T22274 CMB08D 145981960 IC50 > 30000 nM T22274 C2OC6Q 145982084 IC50 = 6.7 nM T22274 CPK9F7 145982364 IC50 = 508 nM T22274 C9VDE5 145982499 IC50 = 2130 nM T22274 CKYP15 145982514 IC50 = 1070 nM T22274 CF8R6Z 145982577 IC50 = 0.2 nM T22274 CY08OG 145982591 IC50 = 71900 nM T22274 CX2LY1 145982614 IC50 = 12220 nM T22274 CHI03D 145982623 IC50 = 0.25 nM T22274 C6QGM5 145982769 IC50 = 2.9 nM T22274 C71AZC 145982856 IC50 = 5.2 nM T22274 CN4T7U 145982897 IC50 = 2.1 nM T22274 CRT9I3 145982975 IC50 = 1780 nM T22274 CA7K6C 145983002 IC50 = 7 nM T22274 CR63YW 145983218 IC50 = 220 nM T22274 CNOG85 145983259 IC50 = 484 nM T22274 C6OL1K 145983267 IC50 = 9750 nM T22274 CE38WZ 145983432 IC50 = 37 nM T22274 CA1LM5 145983443 IC50 = 9 nM T22274 CPUJ75 145983482 IC50 = 3570 nM T22274 CXF9G4 145983559 IC50 = 29 nM T22274 C8O1GU 145983616 IC50 > 10000000 nM T22274 CWD0A9 145983712 Ki = 23 nM T22274 C17UTC 145983813 IC50 = 74400 nM T22274 C2I7EQ 145983818 IC50 = 9040 nM T22274 C34ZQV 145983855 IC50 = 99.3 nM T22274 CV8H2B 145983876 IC50 = 7020 nM T22274 C3I6VL 145983950 IC50 = 320 nM T22274 CJLG54 145984020 IC50 = 1.6 nM T22274 C7FBZ5 145984102 IC50 = 8660 nM T22274 C62UNC 145984122 IC50 = 3.4 nM T22274 CL43AD 145984253 IC50 = 0.85 nM T22274 CIWO70 145984314 IC50 = 9250 nM T22274 C0WBG3 145984326 IC50 = 519 nM T22274 CODK63 145984420 IC50 = 2.3 nM T22274 C9ZKC1 145984665 IC50 = 17300 nM T22274 CX36SR 145984704 IC50 = 5 nM T22274 CXWS04 145984852 IC50 = 9.6 nM T22274 CSA1K8 145984949 IC50 = 6940 nM T22274 C2ND4F 145985023 IC50 = 15.8 nM T22274 CJF71C 145985091 IC50 = 80.8 nM T22274 CT50ZG 145985100 IC50 = 860 nM T22274 CFLH65 145985111 IC50 = 4700 nM T22274 C9MV2L 145985198 IC50 = 300 nM T22274 CN6KB9 145985243 IC50 = 1150 nM T22274 CB24HO 145985400 IC50 > 40000 nM T22274 C60TZP 145985422 IC50 = 2.6 nM T22274 CDM0T5 145985755 IC50 = 13.3 nM T22274 CK90XR 145985933 IC50 = 250 nM T22274 CBF13W 145985947 IC50 = 610 nM T22274 CJV74F 145986075 IC50 = 18.5 nM T22274 C56MWZ 145986208 Ki = 130 nM T22274 CL62QV 145986214 IC50 = 26100 nM T22274 CGN02Q 145986264 IC50 = 210 nM T22274 C51BUM 145986322 IC50 = 1.1 nM T22274 C1WH7V 145986586 IC50 = 420 nM T22274 CS79CE 145986632 IC50 = 709 nM T22274 C7L1GU 145986811 IC50 = 12.6 nM T22274 CFWH51 145987165 IC50 = 41.9 nM T22274 CC12UX 145987331 IC50 = 1970 nM T22274 C2XPR7 145987380 IC50 = 14 nM T22274 CRX8H1 145987492 IC50 = 7 nM T22274 CFH27G 145987566 IC50 = 0.1 nM T22274 CPAX89 145987732 IC50 = 5 nM T22274 CR4YX8 145987935 IC50 = 57 nM T22274 CK6U7Z 145988024 IC50 = 1.3 nM T22274 CV3S8R 145988041 IC50 > 40000 nM T22274 C8XBL4 145988088 IC50 = 3.1 nM T22274 C3GNI6 145988740 IC50 = 968 nM T22274 C82CIN 145988785 IC50 > 30000 nM T22274 C0NI8A 145988806 IC50 = 2.1 nM T22274 C2EXQ1 145989123 IC50 = 60.1 nM T22274 CI97FM 145989333 IC50 = 9.7 nM T22274 CJ8DO3 145989487 IC50 = 78 nM T22274 CX32KW 145989747 IC50 = 444 nM T22274 C5UZ4J 145990125 IC50 = 32 nM T22274 CO4J2D 145990209 EC50 = 20200 nM T22274 CHR0U9 145990400 IC50 = 1.8 nM T22274 C4PSZ2 145990543 IC50 = 40.9 nM T22274 CN1CA2 145990746 IC50 = 584 nM T22274 CO7F1K 145990990 IC50 = 3 nM T22274 C1ZP4A 145991045 IC50 = 679 nM T22274 C8L3XM 145991315 IC50 = 356 nM T22274 CZ94XS 145991731 IC50 = 23 nM T22274 C6WN7O 145992050 IC50 = 203.8 nM T22274 CZ01CR 145992333 IC50 = 1145 nM T22274 CJC47L 145992551 IC50 = 6.1 nM T22274 C3RC5J 145992581 IC50 = 4.6 nM T22274 CD09RT 145992905 IC50 = 1.2 nM T22274 CEP2Q4 145992958 IC50 = 903 nM T22274 C7I5XM 145993519 IC50 = 62.5 nM T22274 C51ZNC 145993585 IC50 = 6.1 nM T22274 CF54BR 145993638 IC50 = 718.6 nM T22274 CF36GI 145993689 IC50 = 6.8 nM T22274 CPSM82 145993919 IC50 = 181 nM T22274 C1W6CF 145994016 IC50 = 110 nM T22274 CSQ7G0 145994254 IC50 = 1.8 nM T22274 C59KOM 146585662 IC50 = 12 nM T22274 CFQO97 146585699 IC50 = 4 nM T22274 C0GMR1 146585718 IC50 = 9 nM T22274 CB7K1M 146676960 IC50 = 31.62 nM T22274 CJYD03 146836277 IC50 = 561.8 nM T22274 CF2YV5 147185900 IC50 = 101 nM T22274 C0YXS8 147254231 IC50 = 56 nM T22274 C3RB5F 147731349 IC50 = 37.95 nM T22274 CA1EC6 147746059 IC50 = 110.4 nM T22274 CV9M5L 147777638 IC50 = 85.35 nM T22274 C7L2GO 147878620 IC50 = 42.98 nM T22274 CKEG86 148044361 IC50 = 21.23 nM T22274 CBG8T7 148123770 IC50 = 43.6 nM T22274 C5KHE1 148150539 IC50 = 15.33 nM T22274 C48EXH 148289288 IC50 = 1406 nM T22274 C3SA6B 148608442 IC50 = 13.6 nM T22274 CT5E1O 148634364 IC50 = 39.07 nM T22274 CWLF12 148743859 IC50 = 20.22 nM T22274 CWCP30 148853853 IC50 = 19531 nM T22274 COH3I8 148951442 IC50 = 50.68 nM T22274 CO47EC 148970856 IC50 = 4.6 nM T22274 C3EFX4 149016806 IC50 = 61.42 nM T22274 CN71OS 149405396 IC50 = 536 nM T22274 CV5ZR0 149819902 IC50 = 22 nM T22274 CH3JE4 150054712 IC50 = 23 nM T22274 C8S3MF 150076000 IC50 = 8.7 nM T22274 C8BM2K 150127738 IC50 = 116.6 nM T22274 C9L7DG 150259632 IC50 = 35 nM T22274 CKMU94 150304623 IC50 = 54.2 nM T22274 CU2XY0 150312795 IC50 = 168 nM T22274 C5PQI9 150470306 Ki = 3.89 nM T22274 C4JP7X 150533939 IC50 = 32 nM T22274 CAQ36F 150619353 IC50 = 24 nM T22274 C89BKD 150622000 IC50 = 4630 nM T22274 C5T1PC 150863979 IC50 = 1455 nM T22274 CIM06Z 150916115 IC50 = 636 nM T22274 CN46CZ 150945374 IC50 = 839.1 nM T22274 CWG10H 151364732 IC50 = 202 nM T22274 CM6IF7 151532669 IC50 = 5 nM T22274 CS0V6U 151543423 IC50 = 57 nM T22274 CV39LB 151825687 IC50 = 1194 nM T22274 CA21YZ 151887635 IC50 = 51 nM T22274 CF7NB5 151976649 IC50 = 15.89 nM T22274 CROU95 152148008 IC50 = 15 nM T22274 CY1NG0 152157103 IC50 = 170 nM T22274 CYF2I5 152375216 IC50 = 20 nM T22274 CL1UA7 152547478 IC50 = 8 nM T22274 C2AOQ6 152562172 IC50 = 10 nM T22274 C6I7OZ 152636346 IC50 = 159 nM T22274 CP6YK7 153056786 IC50 = 56.89 nM T22274 C4F8LC 153265113 IC50 = 97.07 nM T22274 C17DHQ 153406869 IC50 = 33.77 nM T22274 CA17JT 153406872 IC50 = 95.04 nM T22274 CC35YT 153406873 IC50 = 30.89 nM T22274 C0VF5H 153406878 IC50 = 1386 nM T22274 CT4H9P 153408403 Ki = 2.1 nM T22274 CK7P3F 153408410 IC50 = 20 nM T22274 C7LM4U 153534003 IC50 = 780 nM T22274 CP1V9H 153534004 IC50 = 188 nM T22274 C9FIY4 153534005 IC50 = 73 nM T22274 CVT63S 153534008 IC50 > 10000 nM T22274 CW1KJ7 153774772 IC50 = 6280 nM T22274 C7F1UK 155454897 IC50 = 12 nM T22274 CV01JD 155510802 IC50 = 5 nM T22274 C8Q9UG 155510876 IC50 = 27 nM T22274 CIG6K4 155510915 IC50 = 37 nM T22274 C0KW3O 155511274 IC50 > 50000 nM T22274 C0LH8C 155511921 IC50 = 464 nM T22274 CH3UY9 155512029 IC50 = 66 nM T22274 C5K6RO 155512136 IC50 = 32 nM T22274 C2TEZ4 155512242 IC50 = 19 nM T22274 CV2MG0 155512401 IC50 = 46 nM T22274 CQ5BL7 155512551 IC50 > 50000 nM T22274 CGN9Y6 155512914 IC50 = 5.9 nM T22274 CPF6R7 155512997 IC50 = 27.7 nM T22274 C7VKU2 155513116 IC50 > 32000 nM T22274 C5WUJ6 155513192 IC50 = 196 nM T22274 CJ8IQ0 155513281 IC50 = 3.2 nM T22274 CE4H7I 155513471 IC50 > 50000 nM T22274 CN9JW5 155513555 IC50 > 1000 nM T22274 CLY7W3 155513825 IC50 = 12.7 nM T22274 CKQZ35 155514031 IC50 = 198 nM T22274 C6BV9W 155514532 IC50 > 10000 nM T22274 CW3VT9 155514603 IC50 = 9000 nM T22274 CZ84WI 155515284 IC50 > 50000 nM T22274 CA27CY 155515378 IC50 = 1.25 nM T22274 C3IV1T 155515466 IC50 = 17 nM T22274 CWEZ05 155515488 IC50 = 19.66 nM T22274 CUKG21 155515602 IC50 > 50000 nM T22274 C4QLT5 155515638 IC50 = 2670 nM T22274 CAY62H 155515699 IC50 = 37 nM T22274 CR1JH7 155515739 IC50 > 1000 nM T22274 CDM3E7 155515806 IC50 = 18.9 nM T22274 CY2DC1 155515836 IC50 = 13 nM T22274 CYJ53T 155515864 IC50 = 24000 nM T22274 C1K2XN 155516139 IC50 > 50000 nM T22274 C09JPI 155516456 IC50 = 11 nM T22274 CL47DJ 155516579 IC50 = 18130 nM T22274 CA1J3N 155517086 IC50 = 9.7 nM T22274 CL72ME 155517175 IC50 > 50000 nM T22274 C7G0XM 155517418 IC50 > 10000 nM T22274 CYS75R 155517555 IC50 < 0.5 nM T22274 CVI9Y7 155517723 IC50 = 13 nM T22274 CY54TU 155518062 IC50 = 8.2 nM T22274 CEH2N5 155518106 IC50 = 4.4 nM T22274 CE7QS8 155518248 IC50 = 309.4 nM T22274 C58ZNC 155518327 IC50 = 333.33 nM T22274 CMDR68 155518334 IC50 = 63.1 nM T22274 CCDU61 155518496 IC50 > 32000 nM T22274 C41AIO 155518963 IC50 = 151 nM T22274 C86DYH 155519015 IC50 = 115 nM T22274 C5WMN4 155519227 IC50 = 100 nM T22274 CAD06U 155519254 IC50 = 2 nM T22274 CDY5H6 155519645 IC50 = 316 nM T22274 C43HXE 155519794 IC50 = 9 nM T22274 C4P1RM 155520291 IC50 = 3190 nM T22274 C34FXY 155520399 IC50 > 50000 nM T22274 CAD10S 155520741 IC50 > 50000 nM T22274 CC87ZP 155520950 IC50 = 52 nM T22274 CAZ3S7 155521187 IC50 = 11 nM T22274 CZ75FW 155521272 IC50 = 7.6 nM T22274 CG4F2U 155521283 IC50 > 32000 nM T22274 CR7K5H 155521373 IC50 = 592.1 nM T22274 CCV14N 155521717 IC50 = 16 nM T22274 C82PHV 155521822 IC50 > 10000 nM T22274 C6DVZ9 155521965 IC50 > 10000 nM T22274 C0KJ1Z 155522601 IC50 > 50000 nM T22274 CVWC07 155522713 IC50 = 47 nM T22274 CEQ58R 155523224 IC50 = 4.5 nM T22274 C5G6PA 155523673 IC50 = 2527 nM T22274 CJ3E4G 155524660 IC50 > 10000 nM T22274 CBP78G 155524778 IC50 = 215.4 nM T22274 CNW0D1 155524821 IC50 = 2.8 nM T22274 CX6QF0 155524910 IC50 = 10.7 nM T22274 CI24AD 155525662 IC50 > 50000 nM T22274 CN7B1T 155525782 IC50 > 100000 nM T22274 CG1K0O 155526247 IC50 > 50000 nM T22274 COD92I 155526258 IC50 = 132 nM T22274 CV8J0O 155526623 IC50 = 31.1 nM T22274 CGAF52 155526729 IC50 = 12.6 nM T22274 CEB3D1 155526858 IC50 = 16.5 nM T22274 C63NOC 155527045 IC50 = 314 nM T22274 CEM0A3 155527290 IC50 > 50000 nM T22274 CW2H5R 155527295 IC50 > 10000 nM T22274 C71UNO 155527385 Ki = 100 nM T22274 CX12MK 155527651 IC50 = 6 nM T22274 CQK19H 155527955 IC50 > 10000 nM T22274 C61PZK 155528318 IC50 = 540 nM T22274 C7SPF3 155528334 IC50 = 20.5 nM T22274 CHR4K5 155528532 IC50 = 25096.3 nM T22274 CQ4RG3 155528629 IC50 = 14 nM T22274 C0IC6W 155528706 IC50 = 3.1 nM T22274 CK67EB 155529012 IC50 = 9.09 nM T22274 CZ70PO 155529066 IC50 > 50000 nM T22274 C49NGT 155529137 IC50 > 50000 nM T22274 C9L6OC 155529247 IC50 = 17 nM T22274 CX2OS7 155529270 IC50 = 14 nM T22274 C95YJA 155529506 IC50 = 190.1 nM T22274 C94BFW 155529690 IC50 > 10000 nM T22274 CZMC49 155530597 IC50 = 0.79 nM T22274 COTR30 155530602 IC50 = 117 nM T22274 C8AZI6 155530932 IC50 > 50000 nM T22274 C47WTL 155531016 IC50 = 5.7 nM T22274 CZG79N 155531159 IC50 > 50000 nM T22274 CVH13A 155531441 IC50 = 6 nM T22274 CN3W5J 155531452 IC50 > 50000 nM T22274 CUC3P1 155531533 IC50 > 10000 nM T22274 CKV01F 155531688 IC50 = 430 nM T22274 CK2UY4 155531957 IC50 = 1800 nM T22274 CV2C8O 155532194 IC50 = 350 nM T22274 C3HDI1 155532640 IC50 = 898.3 nM T22274 C7U1TE 155532903 IC50 = 7 nM T22274 C1F4DU 155533216 IC50 = 550 nM T22274 C8IMN6 155533398 IC50 = 1995.26 nM T22274 CIZ46A 155533876 IC50 = 6 nM T22274 CF69UC 155534005 IC50 = 17 nM T22274 CK6W2Y 155534018 IC50 = 28 nM T22274 C5X7AF 155534057 IC50 = 5 nM T22274 CPE68B 155534222 IC50 = 125.89 nM T22274 C38BKE 155534255 IC50 = 353 nM T22274 C6LB5D 155535084 IC50 = 36 nM T22274 CJH9L4 155535498 IC50 = 110 nM T22274 C91UNV 155535585 IC50 > 10000 nM T22274 CD49QF 155535974 IC50 = 25 nM T22274 CO91WP 155536301 IC50 = 77 nM T22274 CH27XY 155536857 IC50 > 10000 nM T22274 C81KIF 155537008 IC50 > 40000 nM T22274 C2JH0S 155537112 IC50 > 10000 nM T22274 CQV6H0 155537405 IC50 > 50000 nM T22274 C5FRG0 155537455 IC50 > 50000 nM T22274 CTF98X 155537473 IC50 = 4.8 nM T22274 CAG9P4 155537573 IC50 > 50000 nM T22274 C4BHY7 155537857 IC50 = 7 nM T22274 CPQ98F 155538015 IC50 = 8420 nM T22274 CJ86WN 155538082 IC50 = 14.8 nM T22274 CTU3X6 155538087 IC50 = 12 nM T22274 C50EMD 155538313 IC50 > 1000 nM T22274 C63FKN 155538445 IC50 > 10000 nM T22274 C1PFV7 155538765 IC50 > 5000 nM T22274 C69GOV 155538824 IC50 = 11.8 nM T22274 CLD19W 155539311 IC50 = 40 nM T22274 CU6V4Q 155539319 IC50 > 50000 nM T22274 CM5UN4 155539714 IC50 > 50000 nM T22274 CE6G4A 155539837 IC50 = 16.58 nM T22274 C6U0FM 155540189 IC50 = 6900 nM T22274 C6LQT1 155540719 IC50 > 50000 nM T22274 C7B5NU 155541992 IC50 > 10000 nM T22274 CN7E6U 155542755 IC50 = 26 nM T22274 CJ25HV 155542887 IC50 = 19.5 nM T22274 CZY0N4 155543588 IC50 = 16 nM T22274 CKZ9A5 155543845 IC50 = 71.3 nM T22274 C2G1RZ 155544401 IC50 = 2238 nM T22274 CP4L1F 155544459 IC50 = 14000 nM T22274 CPIQ21 155544472 IC50 = 16.7 nM T22274 CJK31W 155544599 IC50 = 13 nM T22274 CNM3P1 155544603 IC50 > 50000 nM T22274 C1VF5A 155544728 IC50 = 20.1 nM T22274 CXR86J 155545078 IC50 > 50000 nM T22274 CCV9J0 155545380 IC50 = 300 nM T22274 C2UN1K 155545446 IC50 = 129 nM T22274 CX7K3O 155545502 IC50 = 14.2 nM T22274 CNVW40 155545626 IC50 = 660 nM T22274 C7YOP9 155545823 IC50 = 470 nM T22274 C1JSY3 155545907 IC50 = 156 nM T22274 C8DQ7U 155546022 IC50 > 50000 nM T22274 C2E5RQ 155546107 IC50 = 12 nM T22274 CF2O4J 155546325 IC50 > 50000 nM T22274 C2YL1D 155546356 IC50 = 10.3 nM T22274 CK45LA 155546486 IC50 = 19.95 nM T22274 C3HB0U 155546555 IC50 = 125.89 nM T22274 CS3GO2 155546558 IC50 = 3.5 nM T22274 C0AU1L 155546632 IC50 > 50000 nM T22274 C8LT4A 155546691 IC50 > 50000 nM T22274 C93ZWM 155546700 IC50 = 79.43 nM T22274 CEF69A 155546817 IC50 = 7.3 nM T22274 CYR1G0 155547046 IC50 = 136 nM T22274 C8LI9N 155547057 IC50 = 335 nM T22274 C1D4PI 155547606 Ki = 120 nM T22274 CN8CY2 155548358 IC50 = 9.8 nM T22274 CTFU61 155549051 IC50 > 40000 nM T22274 C90FBZ 155549087 IC50 > 50000 nM T22274 CCTU12 155549163 IC50 = 362 nM T22274 CE0YL6 155549538 IC50 = 11200 nM T22274 CFA01C 155549905 IC50 = 148 nM T22274 CO6ID4 155550122 IC50 = 63 nM T22274 C8US1B 155550805 IC50 = 25.3 nM T22274 C4Z5JX 155550827 IC50 > 50000 nM T22274 CA03BO 155551057 IC50 = 79.43 nM T22274 C4Q7CM 155551213 IC50 > 10000 nM T22274 C3JQ1N 155551780 IC50 > 10000 nM T22274 CE01AP 155551891 IC50 = 7.5 nM T22274 CEO4J8 155551917 IC50 = 3253 nM T22274 C05ZVG 155552130 IC50 = 128 nM T22274 C46WHP 155552329 IC50 = 230 nM T22274 CS5D0O 155552399 IC50 = 360 nM T22274 CV4Y5B 155552792 IC50 = 1500 nM T22274 CXT8F1 155552802 IC50 > 50000 nM T22274 CMRJ52 155553215 IC50 = 10 nM T22274 C7PBK3 155553376 IC50 = 120 nM T22274 C9N5ZB 155553414 IC50 = 14 nM T22274 CH8L1V 155554197 IC50 > 10000 nM T22274 CGDF76 155554360 IC50 = 8 nM T22274 CC56ED 155554844 IC50 < 0.17 nM T22274 C7L1NI 155554915 IC50 = 62 nM T22274 CXGR50 155555191 IC50 > 30000 nM T22274 C9DPQ1 155555248 IC50 = 31 nM T22274 CT7GW1 155555345 IC50 = 15 nM T22274 CF2H3O 155555451 IC50 = 455 nM T22274 CZ5OP3 155555490 IC50 = 7.98 nM T22274 CM7FN8 155555499 IC50 = 250 nM T22274 CFW90N 155555562 IC50 = 2.43 nM T22274 CE5P4I 155555900 IC50 = 34 nM T22274 C7QTU1 155555957 IC50 > 50000 nM T22274 CWV2Y0 155556131 IC50 > 10000 nM T22274 CIN57Q 155556138 IC50 = 2.57 nM T22274 CS3QA6 155556824 IC50 = 9 nM T22274 C6IL1E 155557199 IC50 > 50000 nM T22274 C0IO1Q 155557341 IC50 = 17 nM T22274 CNM71L 155557418 IC50 > 50000 nM T22274 CJ9FW6 155557777 IC50 = 28.2 nM T22274 CU78QC 155557817 IC50 > 1000 nM T22274 C5G9IR 155558064 IC50 > 40 nM T22274 CJ3MZ1 155558467 IC50 = 52.8 nM T22274 CK10MB 155558549 IC50 = 137 nM T22274 C0RZ7V 155558710 IC50 = 93 nM T22274 C9Q6MF 155558959 IC50 = 107 nM T22274 C6N2VW 155559068 IC50 = 600 nM T22274 C4XLT3 155559072 IC50 = 1.46 nM T22274 CXY3J1 155559133 IC50 = 17 nM T22274 C2IS1E 155559200 IC50 = 3255 nM T22274 C28CVZ 155559279 IC50 = 1.49 nM T22274 CPD50Q 155559583 IC50 = 95 nM T22274 CY3XI1 155559600 IC50 = 86 nM T22274 CC62UI 155559872 IC50 > 10000 nM T22274 CQ46GB 155559916 IC50 = 26 nM T22274 CMD6Q7 155560250 IC50 = 9.7 nM T22274 CB6Q7T 155560517 IC50 > 40 nM T22274 CID3V4 155560946 IC50 = 14170 nM T22274 CEF98M 155561163 IC50 = 18 nM T22274 CW50YA 155561265 IC50 > 50000 nM T22274 CH0Z1P 155561539 IC50 = 391 nM T22274 C4EQ8P 155561585 IC50 = 380 nM T22274 CJPL17 155561829 IC50 = 10 nM T22274 CJ4KO7 155562145 IC50 > 50000 nM T22274 CGL24S 155562249 IC50 = 300 nM T22274 CXWU93 155563558 IC50 > 40000 nM T22274 C9UYZ6 155564157 IC50 = 2863 nM T22274 C4IM1X 155564305 IC50 = 55.2 nM T22274 CX23YB 155564400 IC50 = 1827 nM T22274 CFH0O8 155564436 IC50 = 35.5 nM T22274 CR85ZW 155564587 IC50 > 10000 nM T22274 C8P5ZA 155564733 IC50 = 12.5 nM T22274 CPNA06 155564750 IC50 > 50000 nM T22274 C87JXN 155564870 IC50 = 158.49 nM T22274 CE0U7K 155564881 IC50 = 188 nM T22274 CAG01V 155565290 IC50 = 28 nM T22274 CZDC03 155565491 IC50 = 33 nM T22274 CG65CR 155565674 IC50 = 1700 nM T22274 C3G1JV 155565712 IC50 = 289 nM T22274 C2IVK7 155565738 IC50 = 14.4 nM T22274 CD05RS 155566122 IC50 > 50000 nM T22274 CAP9F2 155566187 IC50 = 3 nM T22274 C8GES7 155566397 IC50 > 40 nM T22274 C4A0RK 155566461 IC50 > 50000 nM T22274 CR1PC6 155566620 IC50 = 13.6 nM T22274 C51BFK 155566644 IC50 > 10000 nM T22274 C04CGS 155567444 IC50 > 50000 nM T22274 CT6Z4H 155567814 IC50 = 1847 nM T22274 CA7B0F 155568022 IC50 = 12580 nM T22274 CS03PJ 155568350 IC50 > 50000 nM T22274 CX9V3D 155568494 IC50 = 1980 nM T22274 CF2X0U 155568767 IC50 > 40000 nM T22274 C46XEM 155568884 IC50 = 29 nM T22274 C3W7RP 155569171 IC50 = 19 nM T22274 C5NQK8 155569352 IC50 = 3043 nM T22274 CW5XB4 155569484 IC50 > 30000 nM T22274 C3BAZ5 24861442 IC50 = 50.2 nM T22274 D00GBB 11449246 Ki = 7 nM T22274 D00KFF 9882812 Ki = 4500 nM T22274 D00SEE 11379392 IC50 = 19 nM T22274 D01BCK 23382 IC50 > 100000 nM T22274 D01YBR 44591988 IC50 = 303 nM T22274 D02HVH 11427204 IC50 = 230 nM T22274 D02NWS 279980 Ki = 150 nM T22274 D03HNC 17748273 IC50 = 55000 nM T22274 D03QOD 239512 IC50 = 11000 nM T22274 D04DOL 25032059 IC50 = 5 nM T22274 D04KQF 6675804 Ki = 0.9 nM T22274 D04UVL 1133083 IC50 > 50000 nM T22274 D05OVV 11993691 IC50 = 6 nM T22274 D05QBX 44369352 IC50 > 100000 nM T22274 D06FAK 46918725 IC50 = 41 nM T22274 D07MYE 5355635 IC50 = 22 nM T22274 D07YZZ 5173 Ki = 14.5 nM T22274 D08XMS 44591267 IC50 = 9 nM T22274 D09RKA 72946782 IC50 = 433 nM T22274 D09SUO 5269 IC50 > 75000 nM T22274 D0B3ZM 11436024 IC50 = 67 nM T22274 D0E0TA 44454650 IC50 > 50000 nM T22274 D0E9DD 16095101 Ki > 5000 nM T22274 D0G3ZH 25216936 IC50 = 390 nM T22274 D0G6DH 16661454 IC50 = 40 nM T22274 D0H4YW 3611 Ki > 2500 nM T22274 D0K7QR 45269423 IC50 = 20 nM T22274 D0L7HP 6675803 Ki = 2200 nM T22274 D0M1ZI 16095112 IC50 > 50000 nM T22274 D0M9LJ 44454415 IC50 > 50000 nM T22274 D0MC9C 50908800 IC50 = 26 nM T22274 D0MD7H 44454143 IC50 > 50000 nM T22274 D0N9AK 44138031 IC50 = 661 nM T22274 D0Q2GM 44454416 IC50 > 50000 nM T22274 D0Q4AV 25216938 IC50 = 490 nM T22274 D0Q4EG 4882 IC50 = 5540 nM T22274 D0Q5DI 71462653 IC50 = 3.8 nM T22274 D0Q5MC 24753719 IC50 = 2900 nM T22274 D0Q9PO 16095114 Ki = 2000 nM T22274 D0R3XO 44437883 IC50 = 430 nM T22274 D0R7JA 53344908 IC50 = 2300 nM T22274 D0R8JK 25216937 IC50 = 1500 nM T22274 D0T0SK 44138032 IC50 = 124 nM T22274 D0T4JQ 264 IC50 > 2000000 nM T22274 D0T8AJ 23634372 IC50 = 1100 nM T22274 D0U8FC 759408 IC50 > 50000 nM T22274 D0V1HA 24880249 IC50 = 82000 nM T22274 D0W1PV 6918328 Ki = 123.4 nM T22274 D0X4VO 44359538 IC50 = 4300 nM T22274 D0XU0G 44591342 IC50 = 710 nM T22274 D0XZ9Q 11149404 IC50 = 70 nM T22274 D0YP4F 10383069 IC50 = 3 nM T22274 D0Z6MI 44437868 IC50 = 404 nM T22274 D0Z8PX 24757913 IC50 = 1850 nM T49507 D03ZBT 11626560 IC50 > 10000 nM T49507 D09XZB 123631 IC50 = 1000 nM T49507 D0E6XR 3062316 IC50 < 1 nM T49507 D0OB0F 5328940 IC50 = 5.5 nM T49507 D0R0MW 5329102 IC50 > 50000 nM T49507 D0W5HK 216239 IC50 = 0.2 nM T49507 D03LWG 53235510 IC50 > 10000 nM T49507 D04AHQ 71721540 IC50 = 100 nM T49507 D07EHV 44814409 IC50 > 10000 nM T49507 D07HPJ 11476171 IC50 > 10000 nM T49507 D0E3TC 44259 IC50 = 126.4 nM T49507 D0T3ME 156422 IC50 = 900 nM T49507 C63WLY 89644 IC50 > 10 ug.mL-1 T49507 C5JE2Z 104860 IC50 = 8.9 ug.mL-1 T49507 CI1NA5 159926 IC50 > 10 ug.mL-1 T49507 CYBA43 177458 IC50 > 10 ug.mL-1 T49507 CTFM41 777124 IC50 = 76000 nM T49507 CESZ56 938979 IC50 = 300 nM T49507 CN0X9U 3069971 IC50 = 1500 nM T49507 CCN9D5 3142817 IC50 = 610 nM T49507 C4F9UD 3818114 IC50 = 1600 nM T49507 CO6Z9B 4886490 IC50 = 3300 nM T49507 CFW19M 5329009 IC50 = 480 nM T49507 CB23PA 5330197 IC50 = 350 nM T49507 CDQ3M7 5359485 IC50 > 10 ug.mL-1 T49507 C54BYP 5360741 IC50 = 1.4 ug.mL-1 T49507 CS5KX9 9938299 IC50 = 0.4 nM T49507 CUJR40 10062694 EC50 = 4 nM T49507 CVNR70 10254113 IC50 = 4600 nM T49507 C7SFI1 10296883 IC50 > 10000 nM T49507 CQ9C2A 11166116 IC50 = 7100 nM T49507 C28BGP 11177814 IC50 = 190 nM T49507 CD3M4U 11222000 IC50 = 29 nM T49507 CSZ86D 11259287 IC50 = 2200 nM T49507 CLAF52 11259738 IC50 = 230 nM T49507 C6C3JX 11281930 IC50 = 21 nM T49507 C3BE1G 11302787 IC50 = 575 nM T49507 CS98JC 11350978 IC50 = 18 nM T49507 CEV1O4 11398610 IC50 = 389 nM T49507 CF1K8B 11403217 IC50 = 1350 nM T49507 C57TYR 11430707 IC50 = 110 nM T49507 CEM5Q4 11476027 IC50 > 25000 nM T49507 C7P5ZQ 11496099 IC50 = 300 nM T49507 CB0O8F 11497780 IC50 = 138 nM T49507 CGE57U 11504682 IC50 = 402 nM T49507 C7T4CK 11512683 IC50 = 211 nM T49507 C8AY3B 11518031 IC50 < 25 nM T49507 C0RJM4 11525669 IC50 = 165 nM T49507 CL7X4Q 11530963 IC50 = 5100 nM T49507 CG8YW0 11541116 IC50 = 66 nM T49507 C4YOS7 11548082 IC50 = 810 nM T49507 CACS26 11561968 Ki > 2000 nM T49507 C23MSO 11584176 IC50 = 77 nM T49507 CFP2C4 11584673 IC50 = 517 nM T49507 CONZ37 11591872 IC50 = 37 nM T49507 CT54NJ 11606531 IC50 = 518 nM T49507 CSM62L 11626920 IC50 = 672 nM T49507 C23RWH 11670808 IC50 = 158 nM T49507 CPME86 11670863 IC50 = 49 nM T49507 CYA48D 11677791 IC50 = 105 nM T49507 CU0E8O 11690457 Ki > 2000 nM T49507 CJZC08 11692136 IC50 = 850 nM T49507 CB0AP2 11705863 Ki > 2000 nM T49507 CZY05V 11719421 IC50 = 64 nM T49507 CP7AH3 11755812 IC50 = 62 nM T49507 C48PIZ 11756320 IC50 = 69 nM T49507 CDGF78 15282555 IC50 = 3400 nM T49507 C98NES 15980167 IC50 = 84 nM T49507 C67KQF 15980171 IC50 = 2530 nM T49507 CQR5O7 16042971 IC50 > 10000 nM T49507 CQG45C 16109001 IC50 = 8300 nM T49507 C1U8XW 16109036 IC50 = 290 nM T49507 C5JP0A 16407651 IC50 = 14300 nM T49507 COU25S 16420351 IC50 = 8400 nM T49507 C0LZ5T 16663248 IC50 = 36 nM T49507 C6TQ2O 16664354 Ki = 7.27 nM T49507 CZMW48 17377941 IC50 = 8000 nM T49507 CG1YW8 17591826 IC50 = 5200 nM T49507 CCPS81 24764502 IC50 > 35000 nM T49507 CT2M3O 24836812 IC50 = 16000 nM T49507 C39OWF 24836813 IC50 = 240 nM T49507 C5K0GH 24860969 IC50 = 11320 nM T49507 CB62CA 24860971 IC50 = 1550 nM T49507 CTU95J 24861020 IC50 = 5000 nM T49507 CS0Q6V 24861021 IC50 = 1150 nM T49507 CPD28X 24861022 IC50 = 2300 nM T49507 CSF2B4 24861024 IC50 = 1940 nM T49507 CE4L9A 24861026 IC50 = 1330 nM T49507 C2B7GQ 24861075 IC50 = 6000 nM T49507 CV6Y4A 24861080 IC50 = 220 nM T49507 CFK2B9 24882503 IC50 = 430 nM T49507 C0P6AU 24894017 IC50 = 4 nM T49507 CZ6KD4 24894886 IC50 = 44000 nM T49507 CB5TP8 24894992 IC50 = 20000 nM T49507 C32SUJ 24894993 IC50 = 37000 nM T49507 CN13JF 24899915 IC50 = 3.1 ug.mL-1 T49507 CBWR97 24899916 IC50 = 2.1 ug.mL-1 T49507 C9F2JD 24899917 IC50 > 10 ug.mL-1 T49507 C64MTI 24900160 IC50 = 5.9 ug.mL-1 T49507 CO2I6Q 24900161 IC50 > 10 ug.mL-1 T49507 CB79YC 24905143 IC50 = 316 nM T49507 C2DC9J 24905144 IC50 = 4300 nM T49507 CN6V8Z 24905145 IC50 = 220 nM T49507 CSB7P5 24905148 IC50 = 21000 nM T49507 CGSF21 24905149 IC50 > 50000 nM T49507 CVDG02 24905150 IC50 > 50000 nM T49507 CWH6C5 24905152 IC50 = 240 nM T49507 C0HE2Q 24905153 IC50 = 1400 nM T49507 C7QSC9 24905154 IC50 = 2910 nM T49507 CO9D0K 24905155 IC50 = 100000 nM T49507 C5W9UR 24905157 IC50 = 23000 nM T49507 CC1DA3 24905158 IC50 = 17000 nM T49507 COW79F 24905159 IC50 = 100000 nM T49507 CFPA53 24905160 IC50 = 10000 nM T49507 C2O0JX 24905161 IC50 = 100000 nM T49507 CA72BE 24905162 IC50 = 18000 nM T49507 CQN6X9 24905163 IC50 = 22000 nM T49507 CD4O1F 24905165 IC50 = 100000 nM T49507 CKL48T 24905166 IC50 = 100000 nM T49507 C76VYL 24905167 IC50 = 13000 nM T49507 C7K5PU 24905168 IC50 = 2980 nM T49507 CZ57ID 24905169 IC50 = 628 nM T49507 C2DHX9 24905170 IC50 = 100000 nM T49507 CSB96E 24905171 IC50 = 100000 nM T49507 CWZ0R2 24905172 IC50 = 6760 nM T49507 CY3B6M 24905175 IC50 = 244 nM T49507 CW7UA3 24905176 IC50 = 1760 nM T49507 CW1V0H 24905177 IC50 = 760 nM T49507 CO6Y0L 24905178 IC50 = 1100 nM T49507 C60NQW 24905179 IC50 = 1090 nM T49507 C4MO8B 24905180 IC50 = 566 nM T49507 COJI47 24905181 IC50 = 1020 nM T49507 CS0B2C 24905182 IC50 = 96 nM T49507 C1H4BT 24905183 IC50 = 45 nM T49507 C4WHK9 24905184 IC50 = 3300 nM T49507 C7Q4MZ 24905185 IC50 = 353 nM T49507 CS4IP1 24905186 IC50 = 17 nM T49507 C69QWO 24905187 IC50 = 871 nM T49507 C85ANB 24905188 IC50 = 230 nM T49507 CNHD75 24905189 IC50 = 1500 nM T49507 C9JUO2 24905190 IC50 = 2900 nM T49507 CPR03K 24905191 IC50 = 1600 nM T49507 CTAG19 24905193 IC50 = 105 nM T49507 C7VJM5 24905194 IC50 = 3000 nM T49507 CEP1L3 24905195 IC50 = 675 nM T49507 CP68ZD 24905196 IC50 = 380 nM T49507 C8Z0RJ 24905197 IC50 = 1250 nM T49507 CN9RT0 24905198 IC50 = 11000 nM T49507 CHI78P 24905200 IC50 = 1700 nM T49507 CO6PE8 24905201 IC50 = 290 nM T49507 CZ63HS 24905202 IC50 = 340 nM T49507 C2X0FC 24905203 IC50 = 1600 nM T49507 C0WCE3 24905204 IC50 = 10000 nM T49507 CNK50B 24905205 IC50 = 2700 nM T49507 C12DPB 24905206 IC50 = 1400 nM T49507 C8N0RH 24905207 IC50 = 1100 nM T49507 CYA5G2 24905208 IC50 = 2700 nM T49507 CDV2B4 24905209 IC50 = 5000 nM T49507 CEFK68 24905210 IC50 = 2900 nM T49507 CUFP12 24905211 IC50 = 660 nM T49507 C0JG8L 24905212 IC50 = 170 nM T49507 CQ13ZI 24905215 IC50 = 12000 nM T49507 C6VI8F 24905216 IC50 = 3200 nM T49507 CXNH25 24905217 IC50 = 12000 nM T49507 C2PN9S 24905218 IC50 = 32000 nM T49507 C9O2AL 24905219 IC50 = 3800 nM T49507 CIT7U8 24905220 IC50 = 2500 nM T49507 CMD26S 24905221 IC50 = 100000 nM T49507 C4R8WC 24905222 IC50 = 2200 nM T49507 C47SHA 24905223 IC50 = 2300 nM T49507 C1DY2R 24905224 IC50 = 2000 nM T49507 CS0XF9 24905225 IC50 = 100000 nM T49507 CG5VX2 24905226 IC50 = 12000 nM T49507 C57QEO 24905227 IC50 = 100000 nM T49507 C7CG5E 24905228 IC50 = 87000 nM T49507 CHP5D1 24905229 IC50 = 8600 nM T49507 CXP09S 24905230 IC50 = 18000 nM T49507 CY7XG1 24905231 IC50 = 17000 nM T49507 C7JFQ2 24905232 IC50 = 18000 nM T49507 C2JM1P 24905233 IC50 = 14000 nM T49507 CC3BF0 24905234 IC50 = 100000 nM T49507 CE57FI 24905235 IC50 = 7100 nM T49507 CUP20O 24905236 IC50 = 12000 nM T49507 CLC6Q2 24905237 IC50 = 14000 nM T49507 C9M1GI 24905238 IC50 = 15000 nM T49507 CVD72F 24905239 IC50 = 1300 nM T49507 CK38IZ 24905240 IC50 = 5000 nM T49507 CO2V5E 24905241 IC50 = 17000 nM T49507 CZBA19 24905244 IC50 = 4500 nM T49507 CQ8OI1 24905246 IC50 = 100000 nM T49507 CIF2J5 24905251 IC50 = 2630 nM T49507 CPTE58 24905252 IC50 = 27200 nM T49507 CP50RD 24905280 IC50 = 166 nM T49507 CG13ZM 24905281 IC50 = 764 nM T49507 CF0S6X 24905282 IC50 = 4450 nM T49507 C5HBL0 24905284 IC50 = 12200 nM T49507 C2Z5DN 24905285 IC50 = 18300 nM T49507 CL6GH8 24905286 IC50 = 38100 nM T49507 CKYO98 24905287 IC50 = 249 nM T49507 CRNQ65 24905288 IC50 = 737 nM T49507 COD7I5 24905289 IC50 = 1020 nM T49507 C4LP7E 24905290 IC50 = 8930 nM T49507 CE9JC2 24905291 IC50 = 7280 nM T49507 C2GI1R 24905292 IC50 = 100000 nM T49507 CHW8C4 24905293 IC50 = 2520 nM T49507 CQF0H1 24905294 IC50 = 258 nM T49507 CNO7X0 24905295 IC50 = 106 nM T49507 C5WRG7 24905296 IC50 = 456 nM T49507 CQ1S0U 24905297 IC50 = 100000 nM T49507 C4UES7 24905298 IC50 = 100000 nM T49507 CMS69P 24905299 IC50 = 100000 nM T49507 CC0U5M 24905300 IC50 = 18 nM T49507 CW7X6S 24905301 IC50 = 100000 nM T49507 C97IQV 24905302 IC50 = 64 nM T49507 CSJ47V 24905303 IC50 = 7270 nM T49507 CPN74C 24905304 IC50 = 8050 nM T49507 C5CS3N 24905305 IC50 = 352 nM T49507 CK4XE9 24905307 IC50 = 18700 nM T49507 CTU6Z3 24905308 IC50 = 100000 nM T49507 C9SQX1 24905309 IC50 = 492 nM T49507 CM75JP 24905310 IC50 = 100000 nM T49507 C9Q2BJ 24905311 IC50 = 100000 nM T49507 C9VUA1 24905312 IC50 = 468 nM T49507 CU3RS1 24905313 IC50 = 3600 nM T49507 CV5Q7O 24905315 IC50 = 54 nM T49507 C8SA3O 24905316 IC50 = 166 nM T49507 CI5MN3 24905317 IC50 = 256 nM T49507 CJ1P7K 24905318 IC50 = 519 nM T49507 C1T6YQ 24905319 IC50 = 882 nM T49507 CAU86X 24905320 IC50 = 611 nM T49507 C54ISY 24905321 IC50 = 1000 nM T49507 C2GE5I 24905322 IC50 = 1000 nM T49507 C8D6YK 24905323 IC50 = 100000 nM T49507 C5NZH9 24905324 IC50 = 10000 nM T49507 C9D6JR 24905325 IC50 = 2000 nM T49507 CLZT41 24905326 IC50 = 1500 nM T49507 CW8FD3 24905327 IC50 = 254 nM T49507 CHB7A2 24905328 IC50 = 13000 nM T49507 CA8EI3 24905329 IC50 = 100000 nM T49507 CCQ0O7 24905330 IC50 = 1180 nM T49507 CJ81AS 24905331 IC50 = 5800 nM T49507 C8PW4H 24905332 IC50 = 322 nM T49507 C2Y5TF 24905333 IC50 = 347 nM T49507 CH9FL5 24905334 IC50 = 19000 nM T49507 C1S0PC 24905335 IC50 = 17000 nM T49507 C8N9MV 24905336 IC50 = 100000 nM T49507 C9E8BJ 24905338 IC50 = 15000 nM T49507 CX85AC 24905341 IC50 = 100000 nM T49507 CKZ80E 24905342 IC50 = 251 nM T49507 CO8SH1 24905343 IC50 = 3500 nM T49507 C7IZL6 24905344 IC50 = 100000 nM T49507 C7MX9J 25011728 IC50 = 40 nM T49507 CBK82P 25011729 IC50 = 90 nM T49507 C2XB3P 25011730 IC50 = 794 nM T49507 CK47QX 25011731 IC50 = 580 nM T49507 C6GC3X 25014511 IC50 = 3 nM T49507 CYWV64 25014596 IC50 = 32 nM T49507 CB76QL 25014598 IC50 = 8 nM T49507 C64NOS 25014684 IC50 = 7 nM T49507 CN3FQ5 25014760 IC50 = 2 nM T49507 C3WX2S 25014762 IC50 = 17 nM T49507 C3SE8L 25014843 IC50 = 6 nM T49507 CV0RN4 25014844 IC50 = 10 nM T49507 CZ8LP3 25014846 IC50 = 8 nM T49507 CO0R9B 25014936 IC50 = 19 nM T49507 CRA79I 25015025 IC50 = 2 nM T49507 CGDP84 25015026 IC50 = 2 nM T49507 CSD14Z 25015027 IC50 = 35 nM T49507 C0HVE3 25015107 IC50 = 10 nM T49507 C96YKB 25015411 IC50 = 8 nM T49507 CYM80G 25015412 IC50 = 459 nM T49507 CV67GQ 25015556 IC50 = 12 nM T49507 C0TL3X 25015691 IC50 = 28 nM T49507 C0YIC4 25015692 IC50 = 4 nM T49507 CQW9V7 25015693 IC50 = 16 nM T49507 C9RSX2 25015694 IC50 = 10 nM T49507 C3G4VD 25015695 IC50 = 6 nM T49507 C01CUA 25023836 IC50 = 2960 nM T49507 CI4FT9 25023837 IC50 = 2540 nM T49507 CL2X8U 25023838 IC50 = 13960 nM T49507 CU1H8B 25023839 IC50 = 460 nM T49507 CR92ON 25023840 IC50 = 1600 nM T49507 CH7Y6M 25023841 IC50 = 3880 nM T49507 C1FM5R 25023842 IC50 = 640 nM T49507 CGEL03 25023843 IC50 = 20490 nM T49507 C6KL7F 25023844 IC50 = 550 nM T49507 CIV7M4 25023845 IC50 = 1250 nM T49507 CWB47S 25023846 IC50 = 35500 nM T49507 CE93AG 25023847 IC50 = 300 nM T49507 CBW4X9 25023848 IC50 = 41000 nM T49507 CIKU92 25023849 IC50 = 630 nM T49507 CKM2C4 25023850 IC50 = 7850 nM T49507 C02OHK 25023851 IC50 = 1000 nM T49507 C2ICS7 25065806 IC50 = 30 nM T49507 CIH9U3 25114551 IC50 = 14 nM T49507 CFKH56 25114553 IC50 = 15 nM T49507 C6BWZ8 25145145 IC50 = 770 nM T49507 C78YWA 25145716 IC50 = 390 nM T49507 CIG4H0 25178539 IC50 = 2300 nM T49507 C4GI6J 25178540 IC50 = 3900 nM T49507 CS3HT2 25191022 IC50 = 2 nM T49507 CP0K2X 27370767 IC50 > 10000 nM T49507 CJ5U1X 42639664 IC50 = 4.2 ug.mL-1 T49507 C3BH6W 42645046 IC50 = 5 nM T49507 CQ2G4E 42645048 IC50 = 2.6 nM T49507 CKO7F0 42645244 IC50 = 13 nM T49507 C0C1HL 42645248 IC50 = 6 nM T49507 CUR29X 42645268 IC50 = 432 nM T49507 CS3AI0 42645478 IC50 = 2 nM T49507 CTN41Y 44156909 IC50 > 10000 nM T49507 CN0X1C 44156917 IC50 > 10000 nM T49507 C8QF1Z 44198943 IC50 > 10000 nM T49507 C8B3VJ 44198946 IC50 > 10000 nM T49507 CJ1U4M 44199065 IC50 > 20000 nM T49507 CVAU95 44199066 IC50 > 20000 nM T49507 C41DEH 44199068 IC50 = 5400 nM T49507 C8E0LB 44438782 IC50 > 25000 nM T49507 CRZ17Q 44438791 IC50 > 25000 nM T49507 CGI2W1 44438804 IC50 = 3900 nM T49507 CTKD08 44438805 IC50 > 23000 nM T49507 C4Z2VK 44438812 IC50 = 20 nM T49507 CQWC12 44438817 IC50 = 14 nM T49507 C8S3CM 44478400 IC50 = 558 nM T49507 CSQR51 44478936 IC50 = 47 nM T49507 CX3N4F 44478938 IC50 = 1600 nM T49507 C58WTJ 44478939 IC50 = 691 nM T49507 CT4Q0R 44479208 IC50 > 20000 nM T49507 CCG1T2 44479474 IC50 > 20000 nM T49507 C1US6I 44479714 IC50 > 10000 nM T49507 CNYC13 44479715 IC50 > 10000 nM T49507 C4IB1N 44479718 IC50 = 368 nM T49507 CV9IT8 44479956 IC50 = 1200 nM T49507 C59HEM 44479957 IC50 = 236 nM T49507 C3VRO9 44557921 IC50 > 10000 nM T49507 C8AMX5 44564862 IC50 = 1400 nM T49507 CTR59U 44564863 IC50 > 10000 nM T49507 C9EY4C 44564864 IC50 = 800 nM T49507 CG5Z7T 44564910 IC50 = 1000 nM T49507 CU9O4C 44564911 IC50 > 10000 nM T49507 CXZ15S 44564954 IC50 > 10000 nM T49507 CZ78WJ 44564955 IC50 = 3300 nM T49507 CJ1X9V 44565013 IC50 > 10000 nM T49507 CN2Q3D 44565014 IC50 = 780 nM T49507 CM2GN3 44565015 IC50 > 10000 nM T49507 C6RV9I 44565016 IC50 = 840 nM T49507 C23ONL 44581114 IC50 = 209 nM T49507 C0C4NI 44581115 IC50 = 12 nM T49507 CLDY89 44581116 IC50 = 23 nM T49507 C0EY3V 44581117 IC50 = 2 nM T49507 CKJY50 44581142 IC50 = 1 nM T49507 CF47TK 44581143 IC50 = 2 nM T49507 CY3R0L 44581144 IC50 = 7175 nM T49507 CK17IT 44581145 IC50 = 370 nM T49507 CF7W1C 44581173 IC50 = 13 nM T49507 C2SQ3L 44581174 IC50 = 77 nM T49507 C5BC7V 45483150 IC50 = 5000 nM T49507 CH5VI6 46186825 IC50 = 26 nM T49507 CSV9H7 46878646 IC50 = 50000 nM T49507 C6VRE4 46878647 IC50 = 7800 nM T49507 C3Y2IQ 46878648 IC50 = 206 nM T49507 CP6NB8 46878649 IC50 = 744 nM T49507 CE2NP0 46878686 IC50 = 50000 nM T49507 CGS3K5 46878688 IC50 = 2400 nM T49507 CZR3S4 46878689 IC50 = 2100 nM T49507 CQ02DZ 46878690 IC50 = 50000 nM T49507 CS8P7X 46878731 IC50 = 5700 nM T49507 CC63JW 46878732 IC50 = 5400 nM T49507 CY5A9M 46878733 IC50 = 5300 nM T49507 C7H1RG 46878734 IC50 = 6800 nM T49507 C56IYC 46878735 IC50 = 11100 nM T49507 C1J4LY 46878784 IC50 = 50000 nM T49507 CPA61Q 46878844 IC50 = 2900 nM T49507 CV3YQ9 46878845 IC50 = 1700 nM T49507 CJ82NI 46878942 IC50 = 213 nM T49507 C0U8KP 46878943 IC50 = 1700 nM T49507 CA62TK 46878989 IC50 = 1200 nM T49507 C8ATZ0 46878990 IC50 = 1900 nM T49507 C8ZPN4 46878991 IC50 = 10500 nM T49507 CB52HV 46879084 IC50 = 7400 nM T49507 CJ2A3C 46879086 IC50 = 7900 nM T49507 CE7SY4 46879191 IC50 = 938 nM T49507 COGR02 46879192 IC50 = 101 nM T49507 CLHK75 46879291 IC50 = 5700 nM T49507 CM7LR8 46879292 IC50 = 1900 nM T49507 CKHP19 46879293 IC50 = 2500 nM T49507 CY5UL6 46879323 IC50 = 1800 nM T49507 CW6ZS7 46879324 IC50 = 1000 nM T49507 C5U2ZA 46879325 IC50 = 160 nM T49507 CW57XA 46879350 IC50 = 78 nM T49507 CRUP60 46879351 IC50 = 125 nM T49507 CVW72R 46879388 IC50 = 1200 nM T49507 C60GAV 46929544 IC50 > 8000 nM T49507 CP34VL 46929748 IC50 > 1000 nM T49507 CJ2E9Q 46929857 IC50 > 25000 nM T49507 CVS85M 49831162 IC50 = 1.3 nM T49507 CRA74I 49842779 IC50 > 10000 nM T49507 CAZQ43 51003133 IC50 = 38 nM T49507 CXA03W 52920796 IC50 = 700 nM T49507 CU1P2L 52940797 IC50 = 100000 nM T49507 CSX3Z5 52940902 IC50 = 3500 nM T49507 C16TQI 52941019 IC50 = 21 nM T49507 CT20AQ 52942023 IC50 = 121 nM T49507 CX0SA3 52942113 IC50 = 8600 nM T49507 CDHJ08 52942235 IC50 = 3100 nM T49507 CS95FL 52942251 IC50 = 453 nM T49507 C1XEV2 52943394 IC50 = 3710 nM T49507 CJ0Q7G 52944459 IC50 = 219 nM T49507 C39UCS 52944535 IC50 = 300 nM T49507 C5QO8D 52944677 IC50 = 204 nM T49507 CWPC54 52945348 IC50 = 2050 nM T49507 C4NLX7 52945630 IC50 = 14700 nM T49507 C2COM4 52945646 IC50 = 1760 nM T49507 CAX97I 52945780 IC50 = 227 nM T49507 CXD6T8 52945845 IC50 = 3800 nM T49507 C5KBG1 52946934 IC50 = 913 nM T49507 CA6S5L 52946955 IC50 = 117 nM T49507 CU73JY 52947016 IC50 = 460 nM T49507 C3OPZ2 52948082 IC50 = 11 nM T49507 CTM7N2 52948287 IC50 = 513 nM T49507 CKUP78 52948307 IC50 = 246 nM T49507 CF9Y0L 52949373 IC50 = 186 nM T49507 CSK08H 52949391 IC50 = 42 nM T49507 C0FPI8 52949394 IC50 = 190 nM T49507 CSM1B5 52949395 IC50 = 246 nM T49507 CU1F0H 52949547 IC50 = 13 nM T49507 CXQ2S9 52950190 IC50 = 1160 nM T49507 C6OTY5 53251320 IC50 > 30000 nM T49507 CE8OY2 53317913 IC50 = 100 nM T49507 CZ0BV7 53320342 IC50 > 10000 nM T49507 C2W9OA 53324451 IC50 = 7400 nM T49507 C8NA4L 53384644 IC50 = 8700 nM T49507 C0CFZ2 54582972 IC50 = 14 nM T49507 CT7IE4 54583964 IC50 = 5 nM T49507 C5CP1Z 54584912 IC50 = 7 nM T49507 C47JTI 54586838 IC50 = 10 nM T49507 C87YOZ 56929808 IC50 = 150 nM T49507 C6BPR2 58985201 IC50 > 30000 nM T49507 C1MR8Q 60097495 IC50 > 1000 nM T49507 CUBL90 66545750 IC50 = 300 nM T49507 C1HSE0 67035086 IC50 = 5 nM T49507 CWI6K5 67035106 IC50 > 10000 nM T49507 C38RGB 67035556 IC50 = 2700 nM T49507 CV3HW2 67035568 IC50 = 690 nM T49507 CV63UL 67240318 IC50 > 10000 nM T49507 C8I7GC 68293638 IC50 > 10000 nM T49507 CD56XK 68293660 IC50 > 10000 nM T49507 C1WX6V 71544687 IC50 = 300 nM T49507 C5ZKU7 71546969 IC50 = 50 nM T49507 C1BJP3 71546970 IC50 = 177 nM T49507 CAQF28 71547112 IC50 = 1300 nM T49507 C7ARI9 71547113 IC50 = 68 nM T49507 CDOF43 71547115 IC50 = 182 nM T49507 C7E6YV 71720026 IC50 = 14 nM T49507 C62NQZ 76871916 IC50 = 89 nM T49507 C4CMW1 91933866 IC50 = 5.4 nM T49507 C1XM3E 91933868 IC50 = 20 nM T49507 CAU45T 91971978 IC50 > 30000 nM T49507 C0TP3M 118386867 IC50 = 160 nM T49507 CM74AD 118386870 IC50 = 230 nM T49507 C7P3YW 118386917 IC50 = 720 nM T49507 C72ZVL 118386996 IC50 = 15 nM T49507 C4EON3 118387017 IC50 = 24 nM T49507 CQO7Y4 118387022 IC50 = 21 nM T49507 CID08X 118387040 IC50 = 14 nM T49507 CD5Q8T 118387066 IC50 = 560 nM T49507 C1YV9I 118387083 IC50 = 20 nM T49507 CY6J8B 118402527 IC50 = 170 nM T49507 CJ9RO2 118409751 IC50 = 270 nM T49507 CP84XW 118709757 IC50 = 4400 nM T49507 CL0B7G 118709758 IC50 = 2800 nM T49507 C3KLI5 118723185 IC50 > 100000 nM T49507 C9WGB8 127035904 IC50 = 2900 nM T49507 CV8Q7A 135430397 IC50 = 765 nM T49507 C4DG5F 135505693 IC50 = 37 nM T49507 CTJ48K 135524085 IC50 = 1400 nM T49507 CUT1W7 135524168 IC50 = 1700 nM T49507 CU29YK 135750268 IC50 = 1230 nM T49507 CIPA79 135937899 IC50 > 10000 nM T49507 C12UDA 135947972 IC50 = 628 nM T49507 CN42ZS 135947973 IC50 = 316 nM T49507 CF8AO3 135947974 IC50 = 2700 nM T49507 CW08GJ 135947976 IC50 = 14000 nM T49507 CJN7E2 135947978 IC50 = 1370 nM T49507 CFKH34 135947979 IC50 = 95 nM T49507 C9UW0D 137632355 IC50 = 0.27 nM T49507 CQ7MZ6 137633392 IC50 = 92.59 nM T49507 CSQ87K 137634450 IC50 > 1000 nM T49507 CKL1S0 137635182 IC50 > 1000 nM T49507 C9F5GA 137636582 IC50 = 48.53 nM T49507 C6ESL5 137638961 IC50 = 3.6 nM T49507 CX95WZ 137639923 IC50 = 383.59 nM T49507 CP5Q4H 137642451 IC50 = 9.22 nM T49507 CWB74C 137642729 IC50 > 1000 nM T49507 CAY1L6 137645294 IC50 > 1000 nM T49507 C6DOB5 137645672 IC50 = 613 nM T49507 CPI1C6 137646147 IC50 = 179.6 nM T49507 CN5R6A 137646618 IC50 > 1000 nM T49507 CVZ85B 137647227 IC50 = 170.11 nM T49507 CYH05X 137652479 IC50 = 38.14 nM T49507 C1HT8J 137654707 IC50 = 787.89 nM T49507 C1Q7UO 137657235 IC50 = 4.53 nM T49507 C2VRD0 137658292 IC50 > 1000 nM T49507 C8E4QA 137658885 IC50 = 0.13 nM T49507 CZT18Q 137661519 IC50 = 1.26 nM T49507 COCU58 141538430 IC50 = 73.15 nM T49507 C6Y5NP 145949388 IC50 = 86.65 nM T49507 CB3Z1W 145949428 IC50 = 3.87 nM T49507 CGB21E 145949773 IC50 > 500 nM T49507 CVTZ73 145950013 IC50 = 160.1 nM T49507 C3Q1CR 145950413 IC50 > 500 nM T49507 CKU2J6 145951459 IC50 = 38.52 nM T49507 CO0KI7 145951584 IC50 = 44.52 nM T49507 CWUM46 145952127 IC50 = 216.58 nM T49507 CS5FN6 145952182 IC50 > 500 nM T49507 C0U2SX 145952427 IC50 = 334.72 nM T49507 C1C2KL 145952546 IC50 = 15.34 nM T49507 C1KX3F 145952675 IC50 = 37.78 nM T49507 CWU7J4 145952685 IC50 = 106.84 nM T49507 CY3M1A 145952761 IC50 = 24.92 nM T49507 CETX79 145953187 IC50 > 500 nM T49507 CQO92P 145953233 IC50 = 12.1 nM T49507 C6WB5A 145953633 IC50 = 106.84 nM T49507 C09BOY 145953698 IC50 > 500 nM T49507 C8K3IT 145953806 IC50 > 500 nM T49507 CN59EV 145954386 IC50 > 500 nM T49507 CX94IY 145954428 IC50 > 500 nM T49507 C5Z3NW 145954580 IC50 = 15.46 nM T49507 CHBA54 145954987 IC50 > 500 nM T49507 C4CQI1 145955346 IC50 > 500 nM T49507 CFC1R5 145955514 IC50 = 29.28 nM T49507 CZ1X4T 145956589 IC50 = 93.36 nM T49507 C1Z5BV 145956656 IC50 = 87.24 nM T49507 C5VSC7 145956704 IC50 = 4.71 nM T49507 C0Y2TV 145956729 IC50 > 500 nM T49507 CJ4F8V 145956840 IC50 = 73.43 nM T49507 CPG5X6 145957058 IC50 = 47.96 nM T49507 C7YBO3 145957370 IC50 > 500 nM T49507 CZ6O9G 145957666 IC50 = 7.68 nM T49507 CB4P3U 145957792 IC50 > 500 nM T49507 CMSE06 145957839 IC50 = 321.05 nM T49507 CZM5L3 145959497 IC50 = 26.43 nM T49507 CVZ4Q2 145959877 IC50 > 500 nM T49507 CH3YK9 145960253 IC50 = 491.93 nM T49507 CA9LY3 145960784 IC50 > 500 nM T49507 C1U6NF 145961006 IC50 > 500 nM T49507 CMZN84 145961642 IC50 = 133.73 nM T49507 CCK21X 145962292 IC50 > 500 nM T49507 CY7B2V 145962703 IC50 = 78.92 nM T49507 CR75NT 145963742 IC50 = 7.23 nM T49507 CDNC31 145967951 IC50 = 100 nM T49507 C8YM3U 145971698 IC50 > 500 nM T49507 CBI6C0 145971699 IC50 = 17.48 nM T49507 CAR6T3 145971936 IC50 = 21.35 nM T49507 CDB5N6 145972176 IC50 = 23.55 nM T49507 C8S6VJ 145972201 IC50 > 500 nM T49507 CZ5P0E 145972710 IC50 > 500 nM T49507 CC1F9L 147598461 IC50 = 0.32 nM T49507 CS8BJ7 149949125 IC50 > 1000 nM T49507 CJL17Q 150336955 IC50 = 2.21 nM T49507 C6PG4T 150482255 IC50 = 16 nM T49507 CP9JW5 150533442 IC50 > 1000 nM T49507 C2K9BQ 150746217 IC50 > 1000 nM T49507 CHXZ94 151105657 IC50 = 1.49 nM T49507 CU7T8Y 151363744 IC50 > 1000 nM T49507 C24QHN 152058632 IC50 > 1000 nM T49507 CJ4G3V 152221091 IC50 = 2.13 nM T49507 CJSM72 152346156 IC50 = 28.68 nM T49507 CZ7GT5 152346369 IC50 = 0.16 nM T49507 C3BYG8 153529765 IC50 > 1000 nM T49507 CRE82P 155510352 IC50 = 28.62 nM T49507 C2MD1Q 155513187 IC50 > 10000 nM T49507 C5K1UD 155514779 IC50 = 266.77 nM T49507 C83CSB 155515100 IC50 = 2.99 nM T49507 C1S7AI 155516436 IC50 > 1000 nM T49507 CT6V3O 155519533 IC50 > 1000 nM T49507 C6CPO5 155520481 IC50 > 1000 nM T49507 C7QM2L 155520700 IC50 > 1000 nM T49507 CD2YM4 155523255 IC50 = 3.3 nM T49507 CBP7G1 155524105 IC50 = 96.86 nM T49507 CV9Y3X 155527350 IC50 = 0.25 nM T49507 CXY94L 155534355 IC50 > 1000 nM T49507 C9P3ON 155542000 IC50 = 0.44 nM T49507 CP4KT1 155544904 IC50 > 1000 nM T49507 CFG6Z5 155564309 IC50 > 1000 nM T49507 D03EHM 24905142 IC50 = 190 nM T49507 D05FXD 44478401 IC50 = 1.6 nM T49507 D06HVH 54613583 IC50 > 10000 nM T49507 D06QWO 14824655 IC50 > 10 ug.mL-1 T49507 D0A1CM 5281855 IC50 = 1830 nM T49507 D0C2GE 67161540 IC50 = 1250 nM T49507 D0G3SZ 6918469 IC50 = 9.4 ug.mL-1 T49507 D0H1OK 11562302 Ki = 63.8 nM T49507 D0H2CM 135565635 IC50 = 3400 nM T49507 D0R2WK 16038120 IC50 = 1300 nM T49507 D0X8BU 71718651 IC50 = 4400 nM T04303 D0E3TC 44259 IC50 = 235 nM T04303 C3VRO9 44557921 IC50 > 10000 nM T04303 C67OJG 44588117 Ki = 11900 nM T04303 CK80LJ 67130050 IC50 = 4500 nM T04303 CV63UL 67240318 IC50 > 10000 nM T04303 CHI39S 90292823 IC50 = 1520 nM T04303 C4YWO9 134812845 Ki = 270 nM T04303 CG15PY 134812846 Ki = 51000 nM T04303 C9O8CQ 137348448 Ki = 330 nM T04303 C63TGO 137349551 Ki = 91 nM T04303 C6I5ME 137349552 Ki = 350 nM T04303 CI1E8V 137634241 IC50 = 885 nM T04303 CRC8D2 155489850 Ki = 15000 nM T04303 C2MD1Q 155513187 IC50 > 10000 nM T04303 CG8J5X 155518911 Ki = 180 nM T04303 CAN08J 155534113 Ki = 86 nM T04303 C16JRL 155535406 Ki = 220 nM T04303 C3XR8O 155536206 Ki = 470 nM T04303 CX68YN 155541385 Ki > 100000 nM T04303 CWU67H 155543077 Ki = 450 nM T04303 CD8K3O 155543384 Ki = 290 nM T04303 CUTW39 155546618 Ki = 310 nM T04303 C4E0HB 155546757 Ki = 430 nM T04303 C49UVQ 155547733 Ki = 240 nM T04303 CI2J4O 155551330 Ki = 150 nM T04303 CP2K8O 155554487 Ki = 110 nM T04303 CS8MC1 155562025 Ki = 180 nM T04303 C8UW4P 155562878 Ki = 78 nM T04303 CDP94M 155569521 Ki = 510 nM T23471 D00MIN 657298 IC50 = 2810 nM T23471 D05EJG 6305 IC50 = 2250 nM T23471 D05FTJ 4044 IC50 = 980 nM T23471 D06GDY 43815 IC50 = 20 nM T23471 D08VYV 4168 IC50 = 350 nM T23471 D09XQF 3767 IC50 = 4700 nM T23471 D0AN7B 896 IC50 = 3000 nM T23471 D0B2WJ 3371 IC50 = 1800 nM T23471 D0GY5Z 2244 IC50 = 200000 nM T23471 D0K1XK 3637 IC50 = 900 nM T23471 D0K8KX 5280343 IC50 = 1150 nM T23471 D0MA9N 2955 IC50 = 420 nM T23471 D08CJK 1150 IC50 = 770 nM T23471 D08TRG 11528958 IC50 = 630 nM T23471 D09DXX 71571306 Ki = 316.23 nM T23471 D0RO7A 21450 IC50 = 300 nM T23471 D0C0JT 4495 IC50 = 2100 nM T23471 D0Y3LJ 10264211 IC50 = 1000 nM T23471 CB9CG6 1742 IC50 = 2000 nM T23471 C3Y1EB 69982 IC50 > 5000 nM T23471 C8RBI4 159289 IC50 = 7500 nM T23471 C5KHP9 200601 IC50 > 10000 nM T23471 CR9DI6 278475 IC50 = 700 nM T23471 C1K6EZ 649680 IC50 = 6200 nM T23471 CGIY90 688272 IC50 = 7680 nM T23471 CP8LX1 738453 IC50 > 10000 nM T23471 C6GIE5 745587 IC50 = 500 nM T23471 C2R3SD 772603 IC50 = 800 nM T23471 CZX03Q 829306 IC50 > 10000 nM T23471 CBH0O3 829332 IC50 > 10000 nM T23471 C1IFX4 829335 IC50 > 10000 nM T23471 CTV3M2 852586 IC50 = 1600 nM T23471 C1R0KV 866387 IC50 = 1700 nM T23471 CFU4S6 935390 IC50 = 400 nM T23471 C8BSA4 1115191 IC50 = 970 nM T23471 CNCW78 2762738 IC50 = 90 nM T23471 C9CH5B 2769362 IC50 = 28 nM T23471 CN76XG 2835211 IC50 = 44 nM T23471 CN6G1K 2839272 IC50 = 10100 nM T23471 CQ6S5R 3044368 IC50 = 300 nM T23471 CW6GE5 3172238 IC50 = 3800 nM T23471 C9T0CZ 3957066 IC50 = 50 nM T23471 CYH1O6 3992724 IC50 = 24 nM T23471 C1NK4T 4259863 IC50 = 630 nM T23471 CN7F0Z 4874070 IC50 = 3700 nM T23471 C12DWU 4892642 IC50 = 3500 nM T23471 CGO70L 5337997 IC50 > 5000 nM T23471 C6SY9M 6415548 IC50 = 36 nM T23471 CDNC23 6415825 IC50 > 13000 nM T23471 CBC0J5 6418797 IC50 = 84 nM T23471 CS5KM3 6491981 IC50 = 460 nM T23471 COL0M8 6603903 IC50 > 5000 nM T23471 C4N3UF 6604030 IC50 > 5000 nM T23471 CHL7Y8 6861503 IC50 = 1620 nM T23471 C36VYU 7016092 IC50 = 110 nM T23471 C1ERX3 9554777 IC50 = 430 nM T23471 CDQ83I 9590139 IC50 = 80 nM T23471 C95URV 9713809 IC50 = 150 nM T23471 CY0BN1 9716371 IC50 = 3100 nM T23471 C0X7IY 9784772 IC50 = 1130 nM T23471 C1S9CH 9878798 IC50 = 106 nM T23471 CD41KN 9965495 IC50 = 756 nM T23471 CMN41C 10374115 EC50 = 60000 nM T23471 CEIX12 10422576 IC50 > 13000 nM T23471 CY46QR 11600822 IC50 = 704 nM T23471 C1PLC5 11819901 IC50 = 650 nM T23471 CANI87 12146845 IC50 = 8 nM T23471 CGT58N 12399671 IC50 = 5000 nM T23471 C7VSA0 13664293 IC50 = 359 nM T23471 CCB82L 15133393 EC50 = 5 ug.mL-1 T23471 CZ01RO 15547884 IC50 = 13 nM T23471 CP4DG3 15547885 IC50 = 210 nM T23471 CYQ2L9 15547887 IC50 = 60 nM T23471 C0RMJ8 16071339 IC50 = 3000 nM T23471 CV41ZU 16767976 IC50 = 15000 nM T23471 CC82LY 17354973 IC50 = 6200 nM T23471 CAS3T0 17568547 IC50 = 1400 nM T23471 CT8Y7U 17904246 IC50 > 100 nM T23471 CD1X4V 19696832 IC50 = 40 nM T23471 CCW12Q 20501659 IC50 = 2700 nM T23471 CE74PW 21281445 IC50 = 900 nM T23471 CRB6D9 21824639 IC50 = 96 nM T23471 CHW57E 22662950 IC50 = 200 nM T23471 CD35SR 24766375 IC50 = 4148 nM T23471 CF7D1W 25099135 IC50 = 14000 nM T23471 CC9S5U 28412206 IC50 = 320 nM T23471 C8EK9J 28449746 IC50 = 670 nM T23471 CH61YS 28646773 IC50 = 1200 nM T23471 CLB4Y1 44353001 EC50 = 200000 nM T23471 CT89UX 44353003 EC50 = 330000 nM T23471 C4VP3O 44353014 EC50 = 60000 nM T23471 C8YGL6 44390396 IC50 = 49 nM T23471 C0D8SN 44457042 IC50 = 5500 nM T23471 CY04LQ 44457068 IC50 > 100000 nM T23471 CF7Y9G 44457087 IC50 > 100000 nM T23471 C2CO4B 44457088 IC50 = 58000 nM T23471 C5QJE4 44457119 IC50 = 1800 nM T23471 CCOR14 44457122 IC50 = 1600 nM T23471 CQG9C3 44457140 IC50 = 1800 nM T23471 CGI7L0 44457152 IC50 > 100000 nM T23471 C52AIC 45035495 IC50 = 1400 nM T23471 C9FUW6 45784336 IC50 = 1740 nM T23471 C2P7GT 46703570 IC50 = 1028 nM T23471 C38XFD 49787489 IC50 = 5 nM T23471 CX6GP8 49821488 IC50 = 40 nM T23471 CYB26X 49856007 IC50 = 200 nM T23471 CW9S2C 49856008 IC50 = 1000 nM T23471 CVK14B 49856009 IC50 = 850 nM T23471 CS08WQ 49856010 IC50 = 800 nM T23471 C19OFR 49856187 IC50 = 250 nM T23471 CCBS08 49856188 IC50 = 510 nM T23471 CG9B0D 49856189 IC50 = 200 nM T23471 CG24SF 49856190 IC50 = 300 nM T23471 CK1E2F 49856191 IC50 = 170 nM T23471 C8B1VY 49856192 IC50 = 17 nM T23471 CSA90M 49856193 IC50 = 350 nM T23471 C61HSM 49856375 IC50 = 350 nM T23471 C0VT3Z 49856376 IC50 = 63 nM T23471 CV21GT 49856377 IC50 = 18 nM T23471 C5OQS6 49856380 IC50 = 39 nM T23471 C8EG7S 49856569 IC50 = 580 nM T23471 CYZ6T5 53299884 IC50 > 10000 nM T23471 CVZ25P 53299886 IC50 > 10000 nM T23471 CUG78V 53299887 IC50 = 900 nM T23471 CLK9D7 53299888 IC50 > 10000 nM T23471 CTZ06U 53299889 IC50 > 10000 nM T23471 CX2FT3 53344593 IC50 > 100000 nM T23471 C0FZ9G 53360338 IC50 > 100000 nM T23471 CPH4J9 54147697 IC50 = 10 nM T23471 C5T8NI 56956282 IC50 = 800 nM T23471 CY4WT8 57331330 IC50 > 20000 nM T23471 C7SB3R 57331369 IC50 > 20000 nM T23471 C4ALV1 57331603 IC50 = 8000 nM T23471 C26CYT 57331645 IC50 > 20000 nM T23471 CLX5E7 57331685 IC50 = 10000 nM T23471 CXGV20 59917207 IC50 = 650 nM T23471 C7A8HK 67395483 IC50 = 10 nM T23471 CPK5S1 71462358 IC50 = 870 nM T23471 CXRB52 71568996 IC50 = 600 nM T23471 CO51BK 71568997 Ki = 346.74 nM T23471 CMU9E4 71571305 Ki = 173.78 nM T23471 C82CJN 71661340 IC50 = 4 nM T23471 CP7S0W 71661341 IC50 = 21 nM T23471 COU1K0 71661342 IC50 = 3 nM T23471 CM79HR 71661343 IC50 > 100 nM T23471 CUR31L 71661344 IC50 > 100 nM T23471 CY6A0U 71661345 IC50 > 100 nM T23471 C34LBW 71661346 IC50 = 14 nM T23471 C4ZQU3 71661347 IC50 = 27 nM T23471 CSWP81 71661348 IC50 = 11 nM T23471 CQ2YJ9 71661532 IC50 = 5 nM T23471 C1ORE9 71661533 IC50 = 26 nM T23471 C75RSY 71661535 IC50 = 64 nM T23471 CU6O5G 71661536 IC50 = 24 nM T23471 C5RVH3 71661537 IC50 = 132 nM T23471 C7D8QG 71661538 IC50 = 44 nM T23471 C48IPF 71661539 IC50 = 182 nM T23471 CBI0U3 71664049 IC50 = 6 nM T23471 CZ50SG 71729143 IC50 = 807 nM T23471 C75QSV 71729144 IC50 = 1539 nM T23471 C23YBJ 71729145 IC50 = 1078 nM T23471 CN1HE8 71729146 IC50 = 3876 nM T23471 C9LHO4 71729147 IC50 = 2000 nM T23471 C7LS4Z 71729148 IC50 = 1102 nM T23471 C7CJ5Y 71777699 IC50 = 5 nM T23471 CP92FA 72548693 IC50 = 300 nM T23471 C2ANS9 73345497 EC50 = 35000 nM T23471 C08OZW 74015887 IC50 = 85 nM T23471 C9BKT6 76321673 IC50 > 100000 nM T23471 CX2WK8 76321674 IC50 > 100000 nM T23471 CJ9ZB3 76847022 IC50 > 13000 nM T23471 C4V9XO 83318148 IC50 = 1850 nM T23471 CVK95P 83457246 IC50 = 360 nM T23471 CNO73W 83804677 IC50 = 2029 nM T23471 CQ7IY2 83804722 IC50 = 4771 nM T23471 CM19NK 84663516 IC50 > 10000 nM T23471 CLP8T9 85736686 IC50 = 47 nM T23471 CD2RM3 86684674 Ki = 151.36 nM T23471 CP15AE 89557836 Ki = 501.19 nM T23471 CT4ZP3 89557987 Ki = 371.54 nM T23471 CTW37J 92209191 IC50 > 5000 nM T23471 CA0S1L 101805674 IC50 > 10000 nM T23471 CLE2C7 101805678 IC50 > 10000 nM T23471 C7XBZ2 101902833 IC50 = 213 nM T23471 CFB42I 101902837 IC50 = 94 nM T23471 CZ5NH7 104912277 IC50 = 4680 nM T23471 CVZ6C9 118717004 IC50 = 722 nM T23471 CY81BH 118717005 IC50 = 1404 nM T23471 C5PZU2 118717006 IC50 = 711 nM T23471 CV07XJ 118717007 IC50 = 910 nM T23471 C30MPJ 118717008 IC50 > 10000 nM T23471 CNV2O1 118717009 IC50 > 10000 nM T23471 CIC02F 118717010 IC50 = 1787 nM T23471 C37KBD 118717011 IC50 = 1660 nM T23471 C80DOV 118717012 IC50 = 403 nM T23471 C34XID 118717013 IC50 = 140 nM T23471 CTD48X 118948999 IC50 = 4.6 nM T23471 C4SYL0 118949385 IC50 = 120 nM T23471 C4YWT1 118949632 IC50 = 400 nM T23471 CL4KX1 118950056 IC50 = 27 nM T23471 C07CMZ 118950274 IC50 = 12 nM T23471 C9C7FJ 124221770 IC50 = 25 nM T23471 CCJ0Y8 126648798 IC50 = 78 nM T23471 CX96ZI 126648904 IC50 = 720 nM T23471 COZ95K 126648919 IC50 = 24 nM T23471 C2OF9P 126648929 IC50 = 21 nM T23471 C0LI7U 126648996 IC50 = 30 nM T23471 CR7BT5 126649069 IC50 = 23 nM T23471 CH1V7E 126649120 IC50 = 26 nM T23471 C48KCS 126678812 IC50 = 21 nM T23471 C5XF4M 126678836 IC50 = 26 nM T23471 C87MZT 126678883 IC50 = 26 nM T23471 CFJO62 126678929 IC50 = 160 nM T23471 CW8NK2 126678975 IC50 = 6.7 nM T23471 C6BLP7 126680348 IC50 = 21 nM T23471 C6AC8P 126680363 IC50 = 26 nM T23471 C4EJ9M 127037771 IC50 = 100 nM T23471 CGR14F 127037772 IC50 = 100 nM T23471 C7OWR2 127037773 IC50 = 300 nM T23471 CY4QM9 127037774 IC50 = 100 nM T23471 CV6ML3 127037775 IC50 = 900 nM T23471 CWRH56 127038100 IC50 > 20000 nM T23471 C3NK7V 127038102 IC50 = 10000 nM T23471 CD0G9B 127038103 IC50 = 10000 nM T23471 C3OQ1G 127038116 IC50 = 400 nM T23471 C96DOR 127038350 IC50 = 200 nM T23471 CBV1I2 127038367 IC50 = 7000 nM T23471 CWV50I 127038710 IC50 > 40000 nM T23471 CLU2E5 127039056 IC50 = 500 nM T23471 CTY1G6 127039058 IC50 = 600 nM T23471 C73ATR 127039370 IC50 = 400 nM T23471 C2LXC6 127039373 IC50 = 1000 nM T23471 CO1DV3 127040391 IC50 = 300 nM T23471 CZ2HB4 127041065 IC50 = 1200 nM T23471 C7I8MS 127041371 IC50 = 1000 nM T23471 CNA9U5 127041463 IC50 = 1300 nM T23471 CIF10O 127041688 IC50 = 300 nM T23471 C37HMS 127041695 IC50 = 100 nM T23471 C5MQR9 130365202 IC50 = 6.8 nM T23471 CS9PX8 130365266 IC50 = 8.5 nM T23471 C8NL1H 130365899 IC50 = 250 nM T23471 CKB89T 130365913 IC50 = 290 nM T23471 CB91TR 133663694 IC50 > 5000 nM T23471 CC73UG 134130006 IC50 > 5000 nM T23471 CW3NZ0 134130544 IC50 = 110 nM T23471 C51PRO 134131682 IC50 = 370 nM T23471 CUO75T 134133176 IC50 = 370 nM T23471 C50EOL 134137355 IC50 = 660 nM T23471 C3F8OJ 134137742 IC50 = 54 nM T23471 C40EYZ 134138225 IC50 = 85 nM T23471 CSIQ62 134140156 IC50 = 350 nM T23471 CM1N7C 134148444 IC50 = 2500 nM T23471 CE87FH 134152940 IC50 = 490 nM T23471 CT45HM 134153334 IC50 = 1160 nM T23471 C43MXR 134155275 IC50 = 270 nM T23471 CMH36A 134157152 IC50 = 700 nM T23471 CXE81P 135412163 IC50 = 460 nM T23471 CJN4S3 135451354 IC50 = 12000 nM T23471 CSV04G 135685221 IC50 = 340 nM T23471 CN74JH 135775367 IC50 = 1200 nM T23471 C5O2GU 137637141 IC50 = 120 nM T23471 C41BAI 137643798 IC50 = 145 nM T23471 C9MEO2 137646169 IC50 = 40 nM T23471 CKM32D 137659961 IC50 = 130 nM T23471 CM71UQ 145980766 IC50 = 630 nM T23471 CO5V2T 145981031 IC50 > 13000 nM T23471 C8GHU5 145982118 IC50 = 2900 nM T23471 CZ5HP8 145984365 IC50 = 490 nM T23471 C24VDI 145987194 IC50 = 40 nM T23471 C8NUT7 145987843 IC50 = 200 nM T23471 CM5T8V 145989658 IC50 = 78 nM T23471 C2O4FQ 145989963 IC50 = 470 nM T23471 C8OH2X 145990149 IC50 = 510 nM T23471 C9CKN8 145990826 IC50 = 180 nM T23471 C5F2MS 145992066 IC50 > 13000 nM T23471 CKL14J 145992940 IC50 = 200 nM T23471 CU54WQ 145993444 IC50 = 140 nM T23471 C1L6GJ 145993491 IC50 > 13000 nM T23471 D00RIX 5280443 IC50 = 3800 nM T23471 D05DAG 164682 IC50 = 200 nM T23471 D0B5BG 4578 IC50 > 13000 nM T23471 D0G3TK 5280863 IC50 = 2240 nM T23471 D0H6QL 66644 IC50 = 3000 nM T23471 D0S9UQ 345657 IC50 = 900 nM T23471 D0SY6C 5282073 IC50 = 5790 nM T86052 D07VLY 31703 IC50 = 73000 nM T86052 D0W8WB 2353 IC50 = 37000 nM T86052 D09YDM 24360 IC50 > 300000 nM T86052 D0E3TC 44259 IC50 = 8970 nM T86052 D0U2BH 65064 IC50 = 1000 nM T86052 D0U3EP 445154 IC50 = 85000 nM T86052 D0X9HB 6444403 IC50 = 5000 nM T86052 D0J0JH 5281294 IC50 = 6000 nM T86052 D0Q6YP 23205 IC50 = 4000 nM T86052 CY58BM 1880 IC50 = 36000 nM T86052 C26XBL 2017 IC50 = 8200 nM T86052 C7NC2Q 4234 IC50 = 550 nM T86052 CRL6B3 5388 IC50 = 23000 nM T86052 C8IO5D 5389 IC50 = 4500 nM T86052 CW83BF 5390 IC50 = 2800 nM T86052 CIGO04 7081 IC50 = 21700 nM T86052 CF3PD8 62344 IC50 = 12200 nM T86052 CS57LB 72452 IC50 = 100 nM T86052 CR4QL3 72473 IC50 = 11 ug.mL-1 T86052 C72EAP 82143 IC50 = 9400 nM T86052 C5JE2Z 104860 IC50 > 1000000 nM T86052 CS74HZ 145726 IC50 > 40000 nM T86052 C91HBG 147548 EC50 = 5800 nM T86052 C30DMT 157462 IC50 = 3500 nM T86052 C4IRY2 164676 IC50 = 500 nM T86052 CQ9BN3 189219 IC50 > 80 ug.mL-1 T86052 CFQ37A 199438 IC50 = 18197008.59 nM T86052 C0NB5L 335783 IC50 > 50000 nM T86052 CDW73L 355146 IC50 = 100 nM T86052 CQ1X0B 364000 IC50 = 2000 nM T86052 C3MEX9 374309 IC50 = 4500 nM T86052 C54FBS 374311 IC50 = 3500 nM T86052 C7OVY4 399190 IC50 = 200 nM T86052 CEU7P8 446848 EC50 = 5200 nM T86052 CM2NR3 676310 IC50 = 50000 nM T86052 CGQ3K9 688853 IC50 = 3000 nM T86052 C7QKN6 1861620 IC50 = 7130 nM T86052 CMD68Z 2806019 IC50 = 1000 nM T86052 CI0M8F 3084578 IC50 = 51 nM T86052 C7K1LI 3341847 IC50 = 2000 nM T86052 CD4X6E 3446426 IC50 = 160 nM T86052 CD2L5O 3718834 IC50 = 1300 nM T86052 C6ES7I 4033898 IC50 > 40000 nM T86052 C6X5MN 4246984 IC50 = 3396.25 nM T86052 CWD85H 5190042 IC50 = 6194.41 nM T86052 C1GTY6 5281125 IC50 = 15000 nM T86052 CE32PG 5288693 IC50 = 331131121.5 nM T86052 CF62KN 5378308 IC50 > 200000 nM T86052 C0B2QK 5464074 IC50 = 1320 nM T86052 CH2Z8I 9802860 IC50 = 500 nM T86052 CW02DE 9804187 IC50 = 330 nM T86052 CRB4W0 9808666 IC50 = 65 nM T86052 C4I6DJ 9815088 IC50 > 40000 nM T86052 CY03IF 9815161 IC50 = 1200 nM T86052 C3ZQ9U 9818133 IC50 = 400 nM T86052 C59OSA 9830102 EC50 = 60 nM T86052 CQX6Y4 9837937 IC50 > 400000 nM T86052 CUI1T6 9850360 IC50 = 41 nM T86052 CVG76W 9857287 IC50 = 4000 nM T86052 CV0D8T 9858278 IC50 = 800 nM T86052 CRLS05 9879854 IC50 > 40000 nM T86052 CG58TE 9880131 IC50 = 820 nM T86052 C4MT1J 9880186 IC50 = 2200 nM T86052 C4FG6Z 9883224 IC50 = 24000 nM T86052 CSM71G 9900461 IC50 = 3600 nM T86052 CGC68W 9900935 IC50 = 7800 nM T86052 C86XND 9915945 IC50 = 60 nM T86052 C0LWR5 9918266 IC50 = 3600 nM T86052 C9TCE6 9927531 IC50 = 93 nM T86052 CSAN48 9933483 IC50 = 250 nM T86052 CW9DS1 9944144 IC50 = 11000 nM T86052 CKB6X8 9944584 IC50 = 7400 nM T86052 CK3B1D 9947301 IC50 > 40000 nM T86052 CMA85S 9966216 IC50 = 600 nM T86052 C20LJZ 9966473 IC50 = 130 nM T86052 CA9DL5 9986244 IC50 = 750 nM T86052 CT8N5X 10020774 IC50 = 5400 nM T86052 C2X3LA 10028462 IC50 = 9000 nM T86052 C9JT8I 10056382 EC50 = 80 nM T86052 C6E3CI 10065273 IC50 = 5000 nM T86052 C1RG5K 10119878 EC50 = 18 nM T86052 CQLV86 10120540 EC50 = 60 nM T86052 CFE4S3 10120541 EC50 = 21 nM T86052 CJOK01 10120542 EC50 = 1090 nM T86052 C3I2VB 10120705 IC50 = 210 nM T86052 C3MHG8 10121003 EC50 = 460 nM T86052 C7T8RM 10121143 IC50 = 18 nM T86052 CZ50EJ 10121310 IC50 = 40 nM T86052 C1CRK3 10121335 EC50 = 500 nM T86052 C1A8DB 10131832 IC50 = 22100 nM T86052 CD7ZV3 10131931 IC50 = 19000 nM T86052 CWUC72 10144488 EC50 = 1030 nM T86052 CW8FS3 10145782 IC50 = 97723722.1 nM T86052 C54AGY 10158306 IC50 = 470 nM T86052 CJ5FO3 10159351 IC50 = 380 nM T86052 C14KJB 10163490 IC50 = 250 nM T86052 CM8Y1W 10164700 EC50 = 50 nM T86052 C29VRS 10166451 EC50 = 60 nM T86052 C1G2ED 10166452 EC50 = 80 nM T86052 CLB29K 10167766 EC50 = 100 nM T86052 COLS01 10177790 IC50 = 720 nM T86052 CJ8E3V 10186874 EC50 = 140 nM T86052 C93ZRT 10187727 EC50 = 210 nM T86052 C7WU0T 10188027 EC50 = 20 nM T86052 CQOJ70 10188028 EC50 = 200 nM T86052 CM1GB2 10188763 EC50 = 170 nM T86052 C10FUO 10188764 EC50 = 600 nM T86052 C0GT4M 10209287 EC50 = 270 nM T86052 CN24KB 10210368 EC50 = 2730 nM T86052 CY78CM 10212113 EC50 = 67 nM T86052 CQIB92 10224059 IC50 = 760 nM T86052 CUC61J 10231492 IC50 = 210 nM T86052 C6BWZ0 10231493 EC50 = 2 nM T86052 C8TYR2 10280831 EC50 = 1290 nM T86052 CEYJ76 10280832 EC50 = 1330 nM T86052 C7A3IO 10281328 EC50 = 170 nM T86052 COB6U5 10290907 IC50 > 40000 nM T86052 C1PZH3 10294164 IC50 > 40000 nM T86052 CHL6R7 10303003 EC50 = 90 nM T86052 C10TFJ 10303296 EC50 = 660 nM T86052 CB4D6G 10303368 EC50 = 70 nM T86052 CPL56T 10303830 IC50 = 50 nM T86052 CW2ZU5 10304003 EC50 = 100 nM T86052 CHTB86 10304070 EC50 = 30 nM T86052 C80QAL 10319380 IC50 = 128.82 nM T86052 C1KM6O 10350345 EC50 = 98 nM T86052 C72RAW 10385095 IC50 = 230 nM T86052 CXO82P 10386548 IC50 = 380 nM T86052 CTO53X 10410061 IC50 = 10000 nM T86052 CV37LJ 10417437 IC50 = 3400 nM T86052 CEKN47 10436567 IC50 = 3100 nM T86052 CG2A4X 10458944 IC50 = 28 nM T86052 C84TQH 10501060 IC50 = 1100 nM T86052 CQT5U9 10501880 IC50 = 500 nM T86052 C2NX7R 10509552 IC50 > 20000 nM T86052 C2L7JS 10509575 IC50 = 10000 nM T86052 CN9A0J 10509577 IC50 = 16500 nM T86052 CG51SN 10509578 IC50 = 16500 nM T86052 CFVN56 10509579 IC50 = 34500 nM T86052 C47CQP 10509701 IC50 = 33000 nM T86052 CH0VZ4 10530670 IC50 = 50000 nM T86052 C50EOT 10532479 IC50 > 50000 nM T86052 CLI59Q 10550885 IC50 = 1300 nM T86052 C4U8RH 10556139 IC50 > 50000 nM T86052 CI5Z3S 10556818 IC50 = 13200 nM T86052 C40RCU 10556992 IC50 = 25400 nM T86052 CWT2B4 10557162 IC50 = 27300 nM T86052 C4VOP7 10557313 IC50 > 20000 nM T86052 C2CRD5 10567578 IC50 = 630 nM T86052 CXOK35 10574941 IC50 = 4700 nM T86052 C0QE6B 10580510 IC50 = 18500 nM T86052 C2T9NW 10581043 IC50 = 21000 nM T86052 CC5J1N 10602041 IC50 > 50000 nM T86052 CC3S9K 10602711 IC50 > 50000 nM T86052 C95KPA 10604493 IC50 > 50000 nM T86052 CEI41W 10604919 IC50 = 7000 nM T86052 C1L2KC 10605356 IC50 > 20000 nM T86052 C68ZYB 10625702 IC50 = 2300 nM T86052 C9DF1A 10625796 IC50 > 50000 nM T86052 CC8KI7 10626997 IC50 = 16500 nM T86052 CMT32L 10628995 IC50 = 16000 nM T86052 C6AYI9 10629022 IC50 = 7500 nM T86052 COY7F6 10629156 IC50 = 7800 nM T86052 C8B7KI 10652779 IC50 = 8200 nM T86052 C9I8EM 10673434 IC50 > 20000 nM T86052 C72KBR 10675707 IC50 > 50000 nM T86052 C8YG9Z 10676359 IC50 = 14500 nM T86052 CSKE95 10676360 IC50 = 14500 nM T86052 CU8QM7 10676658 IC50 = 8800 nM T86052 COH40L 10676807 IC50 = 8600 nM T86052 C5I1ZD 10694214 IC50 = 6400 nM T86052 CGF1J4 10695455 IC50 = 15500 nM T86052 C6CWS0 10697254 IC50 = 44000 nM T86052 C6FO3B 10699381 IC50 > 50000 nM T86052 C6TVU9 10700612 IC50 = 130 nM T86052 CTE0J6 10700665 IC50 > 20000 nM T86052 CI78CZ 10720763 IC50 = 18500 nM T86052 CIL98W 10721258 IC50 = 14000 nM T86052 C6GRO8 10745169 IC50 = 17000 nM T86052 CJ5I7X 10747913 IC50 = 7800 nM T86052 CV1DN2 10747914 IC50 = 7800 nM T86052 CHJ95L 10747943 IC50 = 13200 nM T86052 CV03LP 10748161 IC50 > 20000 nM T86052 C2JM0G 10767451 IC50 = 2700 nM T86052 C3B7WJ 10767452 IC50 = 4200 nM T86052 CA3RB7 10768302 IC50 = 33500 nM T86052 CE38GA 10768983 IC50 = 8000 nM T86052 CQGK02 10771147 IC50 = 17300 nM T86052 CUS8G1 10795290 IC50 = 16800 nM T86052 C2I3PS 10815021 IC50 = 4300 nM T86052 CG4FS7 10815829 IC50 > 50000 nM T86052 CXM3Y0 10835296 IC50 = 16200 nM T86052 C2KJG9 10836676 IC50 = 4100 nM T86052 CVX4R9 10838712 IC50 = 1800 nM T86052 C5SMJ8 10839598 IC50 = 3700 nM T86052 CE4I6B 10839601 IC50 = 12000 nM T86052 CO17ZB 10842930 IC50 > 20000 nM T86052 CNP47H 10865836 IC50 = 25000 nM T86052 C0L2CA 10973834 EC50 = 18 nM T86052 C80RTA 11049871 EC50 = 570 nM T86052 CR8SJ0 11174461 IC50 = 11700 nM T86052 C8EA4B 11300200 IC50 > 40000 nM T86052 CN5EY9 11430774 IC50 = 45 nM T86052 CN0SW7 11498464 EC50 = 6910 nM T86052 CL3SI1 11498501 IC50 = 3200 nM T86052 CU2V9T 11498709 EC50 = 146 nM T86052 CTVE76 11523680 IC50 = 87000 nM T86052 CY2J6H 11534942 EC50 = 117 nM T86052 C5KC7O 11541962 EC50 = 1930 nM T86052 CQ1X3L 11556599 EC50 = 167 nM T86052 CE2Y5B 11570708 EC50 = 30 nM T86052 CF75XS 11629087 EC50 = 326 nM T86052 C5K4OA 11654469 EC50 > 20000 nM T86052 C3R8CO 11700099 EC50 = 99 nM T86052 CXK6Y2 11707556 EC50 = 255 nM T86052 CQZ27U 11710200 IC50 = 1300 nM T86052 CGD9H8 11717190 IC50 = 3630 nM T86052 C8SF0B 11717499 IC50 = 36700 nM T86052 CFT12H 11766124 IC50 = 9400 nM T86052 CUAP58 11799329 IC50 > 50000 nM T86052 C4QLF3 11802968 IC50 = 4400 nM T86052 CZ8Y1B 12051262 IC50 = 16000 nM T86052 C2IKC5 14213481 IC50 = 30000 nM T86052 CM14YF 14342261 IC50 = 2500 nM T86052 C06NIO 14573901 IC50 = 30 nM T86052 CKDG54 15162830 IC50 > 50000 nM T86052 CAG65Y 15162831 IC50 > 50000 nM T86052 C6JQ0B 15162834 IC50 = 16500 nM T86052 COS59Q 15360568 IC50 = 1000 nM T86052 CXC9J6 15401781 IC50 = 2500 nM T86052 C9U4ZH 15546886 IC50 = 250 nM T86052 C71VZU 15946399 EC50 = 17100 nM T86052 CIO35X 15946460 EC50 = 13300 nM T86052 CG56EB 16447806 IC50 = 24160 nM T86052 CKB95Q 17757387 IC50 = 12.6 nM T86052 CRHC73 18770479 IC50 = 48.98 nM T86052 CXJL51 18770486 IC50 = 338.84 nM T86052 C29OGC 18770490 IC50 = 3890.45 nM T86052 C21TIF 21074073 EC50 = 2300 nM T86052 C4S3MR 21074074 EC50 = 2300 nM T86052 CFQM82 21074076 EC50 = 600 nM T86052 CGP36S 21074077 EC50 = 1900 nM T86052 CI4JU7 21074078 EC50 = 5800 nM T86052 CAEG79 21074082 EC50 = 2300 nM T86052 CMZ7F6 21074083 EC50 = 2300 nM T86052 C41RQO 21074084 EC50 = 1700 nM T86052 C1ZTO9 21074085 EC50 = 1700 nM T86052 C01JHN 21074086 EC50 = 5700 nM T86052 CUEX42 21074087 EC50 = 4300 nM T86052 C27UPB 21074088 EC50 = 4900 nM T86052 CAH4K7 21074089 EC50 = 5900 nM T86052 CP9W1O 21074090 EC50 = 8100 nM T86052 C3QEJ9 21438227 EC50 = 5200 nM T86052 CY7H2I 24882474 EC50 = 1200 nM T86052 CNUP60 24963052 IC50 > 50000 nM T86052 CBT60V 24963056 IC50 = 1350 nM T86052 C4GJ1P 25016911 IC50 = 20 nM T86052 CLM83X 25028063 EC50 > 50000 nM T86052 C2BDM6 25028064 EC50 > 50000 nM T86052 CI01TM 25028065 EC50 > 50000 nM T86052 CV04IU 25087204 IC50 = 8000 nM T86052 CJ3NH4 25107498 EC50 = 800 nM T86052 C1B0MW 25107500 EC50 = 800 nM T86052 CE13LH 25107502 EC50 > 40000 nM T86052 C7HG3E 25107563 EC50 > 40000 nM T86052 CA2G5J 25107566 EC50 > 40000 nM T86052 C3LCI1 25107568 EC50 = 15000 nM T86052 C98CPJ 25107629 EC50 = 1500 nM T86052 C7D5FL 25107631 EC50 = 4000 nM T86052 CNV3Z7 25107633 EC50 > 40000 nM T86052 C7C9NH 25107700 EC50 = 5000 nM T86052 CYU0L2 25107702 EC50 > 40000 nM T86052 C8AV0C 25107704 EC50 > 40000 nM T86052 CXM4W8 25107765 EC50 = 800 nM T86052 CS37ZE 25107767 EC50 = 1500 nM T86052 C9EG2A 25107769 EC50 > 40000 nM T86052 CKC96E 25107834 EC50 > 40000 nM T86052 C6WRG0 25107836 EC50 > 40000 nM T86052 CIAE39 25107838 EC50 > 40000 nM T86052 C7C4AY 25107899 EC50 > 40000 nM T86052 CPTC72 25107901 EC50 = 15000 nM T86052 C1LU2F 25107903 EC50 > 40000 nM T86052 CP2B8W 25107905 EC50 > 40000 nM T86052 CO39QK 25107958 EC50 = 3000 nM T86052 CF8MH4 25107960 EC50 = 1200 nM T86052 CEX68K 25107962 EC50 > 40000 nM T86052 CQG8D6 25108021 EC50 > 40000 nM T86052 CD6QG1 25108023 EC50 > 40000 nM T86052 CVJ2R4 25108025 EC50 > 40000 nM T86052 C65VTY 25108084 EC50 > 40000 nM T86052 CMO0N4 25108282 EC50 = 25000 nM T86052 CTZR23 25108284 EC50 > 40000 nM T86052 CX8J2Q 25108345 EC50 = 25000 nM T86052 C96LTM 25108347 EC50 = 800 nM T86052 C7NH0J 25108349 EC50 = 800 nM T86052 CGW78U 25108391 EC50 = 5000 nM T86052 C38FMZ 25108393 EC50 = 25000 nM T86052 CZ3Y7I 25108395 EC50 > 40000 nM T86052 CYNP09 25108397 EC50 = 10000 nM T86052 CH90RY 25108458 EC50 > 40000 nM T86052 C5FHM9 25108460 EC50 = 1500 nM T86052 C16OVT 25108462 EC50 > 40000 nM T86052 C6VA4K 25108464 EC50 > 40000 nM T86052 CRP58F 25132570 IC50 = 370 nM T86052 CD67AP 25132916 IC50 = 270 nM T86052 CO4X0A 25132918 IC50 = 220 nM T86052 C9O7FX 25132920 IC50 = 160 nM T86052 CJ8Z6S 25133248 IC50 = 310 nM T86052 CNRC10 25133250 IC50 = 200 nM T86052 C0Q1WG 25133252 IC50 = 400 nM T86052 C7HT2P 25195610 IC50 = 18550 nM T86052 C1NQZ2 25197172 IC50 = 21010 nM T86052 CB27KN 25197279 IC50 = 8010 nM T86052 C9IU1F 25197280 IC50 = 15100 nM T86052 C56ABU 42629115 IC50 = 9000 nM T86052 CKNW61 42629237 IC50 = 4000 nM T86052 C4CV0N 44244026 IC50 > 30000 nM T86052 C3OLD9 44244029 IC50 > 30000 nM T86052 CNV05X 44244030 IC50 > 30000 nM T86052 CW0C4F 44244204 IC50 > 30000 nM T86052 CP7R5L 44244205 IC50 = 6000 nM T86052 CV5E8Q 44244206 IC50 = 13000 nM T86052 C3TUM7 44244375 IC50 > 30000 nM T86052 CSD91Y 44244376 IC50 = 12000 nM T86052 CTI84L 44244377 IC50 > 30000 nM T86052 CW3T5L 44244378 IC50 = 7300 nM T86052 CNL2D9 44244545 IC50 = 3000 nM T86052 CXZ62L 44244547 IC50 = 27000 nM T86052 C1C3YN 44244549 IC50 = 4000 nM T86052 CS3HT6 44244551 IC50 = 30000 nM T86052 CL86GU 44244724 IC50 = 5600 nM T86052 CP7BH3 44244725 IC50 = 150 nM T86052 C7N3KX 44266971 IC50 = 9800 nM T86052 C4QNK9 44320145 IC50 > 100000 nM T86052 C8KM4R 44320147 IC50 > 100000 nM T86052 CZQ71A 44320320 IC50 > 100000 nM T86052 CYOD41 44320400 IC50 = 22100 nM T86052 CKHD46 44320409 IC50 > 100000 nM T86052 CED57U 44320415 IC50 > 100000 nM T86052 C4HN0A 44320435 IC50 > 100000 nM T86052 C8Y3GN 44320437 IC50 > 100000 nM T86052 C83WKT 44320439 IC50 = 300 nM T86052 C7HVN9 44320449 IC50 = 29700 nM T86052 CAB87Y 44320451 IC50 > 100000 nM T86052 CL0RU9 44320453 IC50 = 29400 nM T86052 CNFT75 44320479 IC50 = 6800 nM T86052 C2Y3RV 44320507 IC50 = 46900 nM T86052 CIB9G7 44320521 IC50 > 100000 nM T86052 CET98V 44320523 IC50 > 100000 nM T86052 CJ1A2R 44320551 IC50 = 20700 nM T86052 CJ8ST1 44320553 IC50 = 15100 nM T86052 C6SR5H 44320586 IC50 > 100000 nM T86052 CJ39AV 44320606 IC50 > 100000 nM T86052 C5FSH9 44320608 IC50 > 100000 nM T86052 CCF3O2 44320612 IC50 = 13700 nM T86052 CK0U4A 44320614 IC50 > 100000 nM T86052 CWX3U7 44320624 IC50 > 100000 nM T86052 CS1NT4 44320626 IC50 = 9500 nM T86052 CVRD65 44320628 IC50 > 100000 nM T86052 CIY89R 44320630 IC50 > 100000 nM T86052 CY19KG 44320646 IC50 = 6400 nM T86052 CSA2B4 44320691 IC50 = 90700 nM T86052 CH26GP 44320693 IC50 = 11100 nM T86052 C4V7FK 44320695 IC50 = 10600 nM T86052 CQ3H7B 44320697 IC50 = 18300 nM T86052 CGQS24 44320699 IC50 = 45200 nM T86052 C92FDO 44320722 IC50 = 12100 nM T86052 C7VM5U 44320724 IC50 = 3600 nM T86052 CF24RM 44320726 IC50 = 7300 nM T86052 C84ARF 44320746 IC50 > 100000 nM T86052 C2TR6E 44320748 IC50 = 33900 nM T86052 C2R3KS 44320750 IC50 > 100000 nM T86052 CS5Q9V 44320849 IC50 > 100000 nM T86052 CHQ0K2 44320851 IC50 = 22900 nM T86052 C5I3DH 44320853 IC50 = 18900 nM T86052 CES3O6 44339415 IC50 = 11100 nM T86052 CF5TJ9 44339493 IC50 > 50000 nM T86052 CV57JP 44359149 EC50 = 210 nM T86052 C3IC7J 44359561 IC50 = 12000 nM T86052 C9REH1 44359977 IC50 > 50000 nM T86052 CQCV24 44363137 IC50 = 5000 nM T86052 CXE64S 44363393 IC50 = 3100 nM T86052 CT0EY4 44369895 IC50 = 50000 nM T86052 CIP27C 44369906 IC50 = 4200 nM T86052 CU0I3V 44369908 IC50 = 8700 nM T86052 CYQ7Z9 44369916 IC50 = 70000 nM T86052 C3H0TW 44369918 IC50 > 100000 nM T86052 C6Q8UN 44369940 IC50 > 100000 nM T86052 CCG2A4 44370013 IC50 = 35000 nM T86052 CIKT24 44370021 IC50 > 100000 nM T86052 CTLE38 44370030 IC50 > 100000 nM T86052 C8ZBW7 44370045 IC50 > 100000 nM T86052 C8YJD5 44370054 IC50 = 33000 nM T86052 C62EHR 44370064 IC50 = 67000 nM T86052 CO1RK9 44370067 IC50 > 100000 nM T86052 CUT58V 44370073 IC50 = 20000 nM T86052 CUIG58 44370082 IC50 > 100000 nM T86052 C50KNA 44370084 IC50 = 6700 nM T86052 COV38J 44370085 IC50 = 92000 nM T86052 CF6W8J 44370086 IC50 = 41000 nM T86052 C26QJU 44370118 IC50 = 62000 nM T86052 C5IHN7 44370910 IC50 > 100000 nM T86052 CEO92C 44370922 IC50 > 100000 nM T86052 C9VXF3 44370952 IC50 > 100000 nM T86052 CSB81A 44371051 IC50 = 91000 nM T86052 COW1K7 44371103 IC50 = 33000 nM T86052 C38CYB 44371119 IC50 = 75000 nM T86052 CW96JH 44371120 IC50 = 84000 nM T86052 C0I2NH 44371149 IC50 = 7000 nM T86052 CQ8ML9 44371150 IC50 > 100000 nM T86052 CIX96O 44371167 IC50 = 69000 nM T86052 CVD16J 44371172 IC50 = 68000 nM T86052 C6TNA4 44371180 IC50 = 50000 nM T86052 C3C1VT 44371181 IC50 = 64000 nM T86052 CND06O 44371191 IC50 = 79000 nM T86052 CP91OA 44371195 IC50 > 100000 nM T86052 CN5W0S 44371199 IC50 = 79000 nM T86052 CH0UT9 44371200 IC50 = 1000 nM T86052 C5SZ9Y 44371203 IC50 = 76000 nM T86052 CO63XK 44371213 IC50 > 100000 nM T86052 C4B0XT 44371242 IC50 = 56000 nM T86052 CC5MP3 44371243 IC50 = 64000 nM T86052 CWS4V5 44371508 IC50 = 76000 nM T86052 CZB5X6 44392875 EC50 = 318 nM T86052 CU9CO8 44392876 EC50 = 267 nM T86052 C53WIU 44392877 EC50 = 165 nM T86052 CWOU31 44395686 EC50 = 200 nM T86052 C79RVM 44395702 EC50 = 400 nM T86052 C1C4MX 44395736 EC50 = 700 nM T86052 CEP5X7 44395756 EC50 = 200 nM T86052 CQR93P 44395759 EC50 = 2800 nM T86052 CU0TJ4 44395807 EC50 = 200 nM T86052 CD7LO2 44395808 EC50 = 90 nM T86052 C6IUO1 44395828 EC50 = 1900 nM T86052 CWMH45 44395830 EC50 = 5200 nM T86052 CR29JB 44395888 EC50 = 1900 nM T86052 CUOH89 44421795 IC50 = 60 nM T86052 C0AC3T 44421796 IC50 = 400 nM T86052 C10TQX 44438270 EC50 = 350 nM T86052 CKFP93 44438271 EC50 = 1000 nM T86052 CN0TW5 44438272 EC50 = 240 nM T86052 CAG62V 44438274 EC50 = 860 nM T86052 CYQH13 44438275 EC50 = 880 nM T86052 C7JAE6 44438276 EC50 = 440 nM T86052 C78KQT 44438277 EC50 = 230 nM T86052 CY9T0M 44438278 EC50 = 390 nM T86052 C7S4KD 44438279 EC50 = 360 nM T86052 C6T5ED 44447084 IC50 = 20 nM T86052 CQX4T9 44449504 IC50 = 2.2 nM T86052 CP3Q5J 44459278 IC50 = 140 nM T86052 CY3QT5 44461015 IC50 > 50000 nM T86052 C83RFJ 44461056 IC50 = 2700 nM T86052 CN1KG4 44461088 IC50 = 5800 nM T86052 CWQY53 44461129 IC50 = 8200 nM T86052 CD09FQ 44461224 IC50 = 4400 nM T86052 CMB9F0 44461225 IC50 = 2600 nM T86052 CQD3B5 44461331 IC50 = 5400 nM T86052 C2QW9L 44461370 IC50 = 8000 nM T86052 CT70JP 44461371 IC50 = 4100 nM T86052 C9A8FC 44590879 IC50 = 7500 nM T86052 CA3SN8 44659762 IC50 = 30000 nM T86052 C2W8XC 46883408 IC50 > 50000 nM T86052 CAV4N5 46883445 IC50 = 267 nM T86052 C4WTR6 46898227 IC50 = 46773514.13 nM T86052 CV9QL6 46911061 IC50 = 800 nM T86052 C51ZRI 46911062 IC50 = 18.45 ug.mL-1 T86052 CW23IQ 49797864 IC50 = 46700 nM T86052 CY2QS8 49797865 IC50 = 20900 nM T86052 CDZ70H 49797866 IC50 = 3500 nM T86052 C2C0HO 49797867 IC50 = 2500 nM T86052 C3NHI4 49797885 IC50 = 3100 nM T86052 CEX4S7 50993401 IC50 = 5 nM T86052 CSJ8D9 51348634 IC50 = 4200 nM T86052 C90LAI 51349410 IC50 = 10000 nM T86052 C2H7JR 51349694 IC50 = 10000 nM T86052 C9D4FS 51349696 IC50 = 3000 nM T86052 CA9VE8 52942487 IC50 = 4000 nM T86052 C85ZQL 52943972 IC50 = 6500 nM T86052 C4VE1C 52944765 IC50 = 1800 nM T86052 CX5YW4 52947233 IC50 = 9600 nM T86052 CK4OU9 52950008 IC50 = 29100 nM T86052 CLC15N 53233129 IC50 = 4000 nM T86052 CRM6D9 53298010 IC50 = 899.5 nM T86052 C7HND9 53372364 IC50 > 10000 nM T86052 CF4G7H 53372753 IC50 > 10000 nM T86052 C2E7HZ 53770797 IC50 > 50000 nM T86052 CFKQ69 54450017 IC50 = 13000 nM T86052 CD9Y0F 54582780 IC50 = 16800 nM T86052 C0B1JX 54583763 IC50 = 31500 nM T86052 C5NBI8 54583764 IC50 = 24500 nM T86052 CQ9Y2M 54583765 IC50 = 9500 nM T86052 C2IGV4 54583766 IC50 = 17300 nM T86052 CB7S2T 54584754 IC50 = 12500 nM T86052 C65QOK 56598341 IC50 = 1270 nM T86052 C4ES9G 56598342 IC50 = 2020 nM T86052 CW8YV4 56598343 IC50 = 2450 nM T86052 CG0UY4 56598344 IC50 = 1660 nM T86052 CS0XF7 56598345 IC50 = 1830 nM T86052 C2QX8D 56969926 IC50 = 29300 nM T86052 CT3UA7 56970355 IC50 = 7400 nM T86052 C6M1PO 56970358 IC50 = 7700 nM T86052 CD70VU 57390333 IC50 = 12150 nM T86052 C75BKF 57393865 IC50 = 2710 nM T86052 CTNG35 57393866 IC50 = 3670 nM T86052 CR9J8Y 57395591 IC50 = 3660 nM T86052 CLAS98 57395592 IC50 = 5890 nM T86052 C8C4PU 57395593 IC50 = 15780 nM T86052 CA7TK0 57399076 IC50 = 2930 nM T86052 C1OXC9 57399077 IC50 = 5040 nM T86052 C6P1MD 57399078 IC50 = 4650 nM T86052 C2RAL0 57399079 IC50 = 2440 nM T86052 C3MB6P 57400820 IC50 = 3260 nM T86052 C53SMX 57400821 IC50 = 2340 nM T86052 CWMV38 57402580 IC50 = 8210 nM T86052 CPVT67 57402581 IC50 = 2910 nM T86052 CC8EI2 58405960 IC50 = 5000 nM T86052 CS76JF 58984392 IC50 = 220 nM T86052 C6BTW0 59051884 IC50 = 9110 nM T86052 C86KZF 59051887 IC50 = 5990 nM T86052 C60CIH 59051889 IC50 = 8810 nM T86052 C94FQD 59051890 IC50 = 42120 nM T86052 C8F3DR 59052022 IC50 = 2000 nM T86052 C27USE 59052023 IC50 = 4110 nM T86052 CO8K0U 60148177 IC50 = 6698.85 nM T86052 C8YU5N 71449573 IC50 = 3970 nM T86052 CX30VT 71451383 IC50 = 3120 nM T86052 CE8C4F 71453188 IC50 = 17650 nM T86052 CX1TR5 71453192 IC50 = 3550 nM T86052 C1O8RB 71454933 IC50 = 1540 nM T86052 CF0Y5V 71454934 IC50 = 15030 nM T86052 C36ZMO 71455225 IC50 = 34700 nM T86052 C4T0YA 71456711 IC50 = 12090 nM T86052 CGID71 71456712 IC50 = 1240 nM T86052 C6REX5 71456714 IC50 = 3590 nM T86052 CP08HV 71456715 IC50 = 17120 nM T86052 C67ZRQ 71458553 IC50 = 7880 nM T86052 C2EA8M 71458555 IC50 = 6380 nM T86052 C7TH5I 71458562 EC50 = 4000 nM T86052 C75SPM 71462092 IC50 = 13440 nM T86052 C64DOX 71462397 IC50 = 14500 nM T86052 CS48JE 71520680 IC50 = 780 nM T86052 C9WY8B 71520772 IC50 = 1710 nM T86052 CLQ08P 71520773 IC50 = 10820 nM T86052 CKUP81 71520774 IC50 = 3140 nM T86052 C1E4KM 71520775 IC50 = 6600 nM T86052 C0R1GB 71520776 IC50 = 21900 nM T86052 CDQ7T3 71520777 IC50 = 2110 nM T86052 CZOI95 71520778 IC50 = 14800 nM T86052 C94NGJ 71552358 IC50 = 8700 nM T86052 CKMW67 71552440 IC50 = 18492.69 nM T86052 C95MHU 71552441 IC50 = 25700 nM T86052 COWA68 71552442 IC50 = 23800 nM T86052 CL31HA 71552443 IC50 = 22900 nM T86052 CP16YD 71552444 IC50 = 13396.77 nM T86052 C5XA6Z 71552445 IC50 = 10592.54 nM T86052 C52UGW 71552446 IC50 = 37400 nM T86052 CGM7C9 71552539 IC50 = 68300 nM T86052 CAVC04 71552540 IC50 = 83560.3 nM T86052 CIW32Z 71552541 IC50 = 82603.79 nM T86052 COT27P 71552542 IC50 = 76383.58 nM T86052 CSZF74 71552543 IC50 = 54954.09 nM T86052 C18ZWI 71552544 IC50 = 46665.94 nM T86052 C5I3ZU 71552545 IC50 = 93110.79 nM T86052 CPO9B1 71575241 IC50 = 12800 nM T86052 C6HMR5 71575242 IC50 = 7300 nM T86052 CAOG82 71575243 IC50 = 2800 nM T86052 CIFP54 71575244 IC50 = 800 nM T86052 CA7LG3 71575245 IC50 = 1100 nM T86052 C1LX3V 71575357 IC50 = 3100 nM T86052 CN35MF 71575358 IC50 = 5500 nM T86052 C3G6DL 71575359 IC50 = 3000 nM T86052 C29JMW 71575360 IC50 = 900 nM T86052 CA1VS7 71575361 IC50 = 10800 nM T86052 C63KHF 71575362 IC50 = 9300 nM T86052 C3FLZ4 71575363 IC50 = 5100 nM T86052 CO9N7K 71575469 IC50 = 3100 nM T86052 C4B2MW 71575470 IC50 = 2900 nM T86052 CV18CY 71575471 IC50 = 4800 nM T86052 CV89DY 71720658 IC50 = 7294.58 nM T86052 CN5EY0 72197079 IC50 > 50000 nM T86052 C50PBM 72197614 IC50 = 30900 nM T86052 CAK31E 72197615 IC50 = 2300 nM T86052 CHFI10 73349232 IC50 = 1300 nM T86052 CL97NQ 76285562 IC50 = 2000 nM T86052 C7RMC0 76285871 IC50 = 1820 nM T86052 C6XT3G 76286016 IC50 = 910 nM T86052 C0X4PF 76287666 IC50 = 35660 nM T86052 CZ84MI 76287667 IC50 = 28910 nM T86052 CPI9Y1 76287811 IC50 = 3070 nM T86052 CFM1G4 76287813 IC50 = 19660 nM T86052 C87ZUM 76287814 IC50 = 40300 nM T86052 CNL6G7 76309576 IC50 = 3300 nM T86052 CWEP39 76309577 IC50 = 2187.76 nM T86052 C5RPV4 76309584 IC50 = 56 nM T86052 C8W3DL 76310630 IC50 = 920 nM T86052 C2K5RT 76310633 IC50 = 1040 nM T86052 C78RGM 76310634 IC50 = 4650 nM T86052 CWI50N 76313277 IC50 = 3388.44 nM T86052 CF56NJ 76313278 IC50 = 3400 nM T86052 CQ1O2I 76316818 IC50 = 1000 nM T86052 CGF75U 76316823 IC50 = 220 nM T86052 C9PS0L 76316824 IC50 = 2290.87 nM T86052 CEF02P 76320520 IC50 = 3300 nM T86052 CG6DH5 76320522 IC50 = 1995.26 nM T86052 CPR54I 76320523 IC50 = 740 nM T86052 C3LA2E 76320524 IC50 = 2570.4 nM T86052 C9KPX1 76324163 IC50 = 3300 nM T86052 CLY5S9 76324171 IC50 = 3500 nM T86052 C0OE7X 76324863 IC50 = 470 nM T86052 CFZ78X 76327723 IC50 = 2800 nM T86052 C7SA8X 76327730 IC50 = 300 nM T86052 CIJ93P 76327731 IC50 = 3000 nM T86052 CA4R1P 76328704 IC50 = 8890 nM T86052 CU87OW 76328705 IC50 = 25110 nM T86052 CZH43W 76331386 IC50 = 489.78 nM T86052 CMV65L 76331393 IC50 = 890 nM T86052 CO8LD1 76331394 IC50 = 950 nM T86052 CA58JR 76331395 IC50 = 3388.44 nM T86052 CG30XH 76332389 IC50 = 2000 nM T86052 C52XWM 76332392 IC50 = 1190 nM T86052 CD4LV7 76334985 IC50 = 3388.44 nM T86052 CDM2E7 76334986 IC50 = 2500 nM T86052 CZM4A5 76334988 IC50 = 510 nM T86052 CIKZ32 91538550 IC50 = 10000 nM T86052 CW6U3B 91937021 IC50 = 1900 nM T86052 CIL3D8 91937022 IC50 = 200 nM T86052 CAL9N6 91937023 IC50 = 49000 nM T86052 CV3OB4 102420663 IC50 = 20 nM T86052 C4OT2R 118710797 IC50 = 900 nM T86052 CW9VS6 118710798 IC50 = 600 nM T86052 CE2W9B 118710799 IC50 = 1600 nM T86052 CT40FH 118713215 IC50 = 900 nM T86052 C9JPO1 118713217 IC50 = 3000 nM T86052 C3FT1D 118713219 IC50 = 300 nM T86052 CE5D0I 118713221 IC50 = 1100 nM T86052 CBI8Q0 118713223 IC50 = 100 nM T86052 CY0O6M 118713225 IC50 = 70 nM T86052 CP36NK 118713227 IC50 = 500 nM T86052 CN3AZ9 118713228 IC50 = 80 nM T86052 CZ3MJ6 118718019 IC50 = 20 nM T86052 C0DTW1 118723731 IC50 = 300 nM T86052 C4J3GF 118726887 IC50 = 1980 nM T86052 CC30RJ 118726888 IC50 = 49000 nM T86052 CSWK78 118726889 IC50 = 12200 nM T86052 C4EBX6 118726890 IC50 = 1020 nM T86052 CWB95K 118734726 IC50 = 110 nM T86052 C9KXD7 118734727 IC50 = 340 nM T86052 CL59GT 118734729 IC50 = 15170 nM T86052 CPA79N 118734730 IC50 = 2010 nM T86052 C2E7DQ 118734731 IC50 = 1410 nM T86052 C5UJD2 122197484 IC50 > 50000 nM T86052 CUE1T8 127030072 IC50 = 10970 nM T86052 C2TRX0 127030073 IC50 = 54360 nM T86052 CB7XJ0 127030342 IC50 = 8400 nM T86052 CKA97D 127030381 IC50 = 35720 nM T86052 CDY84P 127030382 IC50 = 31210 nM T86052 C69TSJ 127030687 IC50 = 57790 nM T86052 C34TNZ 127030689 IC50 = 5570 nM T86052 CD3W6L 127030690 IC50 = 3300 nM T86052 CS47ZQ 127030691 IC50 = 4770 nM T86052 CS8Y0X 127030988 IC50 = 3030 nM T86052 C62FAI 127031253 IC50 = 6770 nM T86052 CO09NL 127031348 IC50 = 31270 nM T86052 C7DI3S 127031350 IC50 = 3150 nM T86052 C0U6FN 127031351 IC50 = 6680 nM T86052 CNFG45 127031352 IC50 = 3520 nM T86052 C9J1XW 127031353 IC50 = 9320 nM T86052 C0M3CW 127031837 IC50 = 11850 nM T86052 CD26JU 127031906 IC50 = 2100 nM T86052 CV85EN 127031923 IC50 = 3170 nM T86052 C4SM9G 127031926 IC50 = 980 nM T86052 CI56FS 127031951 IC50 = 29810 nM T86052 C8MQZ6 127032171 IC50 = 4630 nM T86052 CI7DJ3 127032172 IC50 = 5440 nM T86052 C7Q5ZH 127032173 IC50 = 22250 nM T86052 CS7TK5 127032180 IC50 = 9940 nM T86052 CSM7H5 127032417 IC50 = 3680 nM T86052 C6UQ1J 127032458 IC50 = 41180 nM T86052 CE3S0J 127032777 IC50 = 14250 nM T86052 CFA8B9 127032778 IC50 = 2120 nM T86052 CX42MC 127032779 IC50 = 6300 nM T86052 C5JLU2 127032780 IC50 = 5690 nM T86052 CE50FQ 127032781 IC50 = 3540 nM T86052 CQ3GK0 127032782 IC50 = 6200 nM T86052 CT07HN 127032783 IC50 = 1270 nM T86052 C86UGD 127033164 IC50 = 3170 nM T86052 CW3C6Q 127033470 IC50 = 24950 nM T86052 C2PR8T 127033625 IC50 = 18150 nM T86052 C5ANJ8 127033940 IC50 = 3440 nM T86052 CW4LP7 127033941 IC50 = 11030 nM T86052 CS68KW 127033942 IC50 = 8740 nM T86052 CY2TN7 127033944 IC50 = 2270 nM T86052 CE85DK 127034202 IC50 = 13100 nM T86052 CER4O8 127034298 IC50 = 1860 nM T86052 CT6YI8 127034316 IC50 > 60000 nM T86052 CLTM14 127034567 IC50 = 4000 nM T86052 CHS8E4 135430795 IC50 = 8600 nM T86052 C24QNA 135442972 IC50 = 147 nM T86052 C29JME 135985961 IC50 = 2300 nM T86052 COI15R 136035760 IC50 = 18990 nM T86052 CC78DB 136035761 IC50 = 15170 nM T86052 CN4RB2 136203000 IC50 = 2000 nM T86052 CA32PC 136491905 IC50 = 1160 nM T86052 CZT71M 137321735 IC50 = 3000 nM T86052 C3HB4Y 137628882 IC50 = 6000 nM T86052 C3G5VL 137629166 IC50 = 3000 nM T86052 C0QCR2 137629168 IC50 = 12000 nM T86052 C1ZBT6 137635029 IC50 = 30090 nM T86052 C7LW5E 137639711 IC50 = 1730 nM T86052 CQ3B0F 137641707 IC50 = 1650 nM T86052 C1JOP3 137645498 IC50 = 968.9 nM T86052 C6A9YR 137650209 IC50 = 28080 nM T86052 CJ45BA 137659690 IC50 = 1580 nM T86052 CKFO90 145977827 IC50 = 300 nM T86052 COH12T 155523186 IC50 = 1020 nM T86052 CUDR38 155529460 EC50 = 23500 nM T86052 D01BAK 9809446 IC50 = 3100 nM T86052 D04KDW 10719801 IC50 = 2000 nM T86052 D04POR 104794 IC50 = 200 nM T86052 D07KNG 5281437 IC50 = 65000 nM T86052 D0A4EA 445639 IC50 = 8600 nM T86052 D0L8BN 44559995 IC50 > 250000 nM T86052 D0P0WG 3624 IC50 = 2100 nM T86052 D0Q2YJ 6763 IC50 = 500 nM T86052 D0V6DE 5282761 IC50 = 16000 nM T86052 D0X5LN 688798 IC50 = 200 nM T86052 D0X9YD 65036 IC50 = 500 nM T86052 D0Y2RR 10038861 IC50 = 1700 nM T86052 D0YJ3Q 5322065 IC50 > 40000 nM T31514 D04AIT 5280445 IC50 = 5.96 ug.mL-1 T31514 D04ZTY 444020 IC50 = 5600 nM T31514 D0AD5C 41774 IC50 = 817380 nM T31514 D0D0ZD 441314 IC50 = 350 nM T31514 D0HR8Z 51634 IC50 = 100 nM T31514 D0MU9L 176077 IC50 = 6000 nM T31514 D0RE9C 501391 IC50 = 1500 nM T31514 D0S5LT 29435 IC50 = 60 nM T31514 CPU1B4 4381 Ki = 54000 nM T31514 CG16SV 10436 IC50 > 100000 nM T31514 C2T0ZI 68072 IC50 > 100000 nM T31514 CG0YT4 92381 Ki = 420 nM T31514 C8XO2U 162350 IC50 = 68.71 ug.mL-1 T31514 CBJ30L 444254 IC50 = 5000 nM T31514 CN2HT8 445074 IC50 = 300000 nM T31514 C1NL4G 636783 IC50 = 0.25 ug.mL-1 T31514 C2ZT1Q 3238144 Ki = 3700000 nM T31514 CH9TY7 3262578 Ki = 75000 nM T31514 CW8TS1 5315170 IC50 > 100 ug.mL-1 T31514 C0DI5P 6443296 IC50 = 0.16 ug.mL-1 T31514 C9SF7P 9535379 IC50 = 11870 nM T31514 CR65TJ 9815399 IC50 = 402 nM T31514 CW3P0D 9880776 IC50 = 3400000 nM T31514 CJ6TV8 10011928 IC50 > 1000000 nM T31514 C0VWI8 10039088 Ki = 1000 nM T31514 CZT1D2 10080697 Ki = 29400 nM T31514 CT2CI5 10548301 IC50 > 100000 nM T31514 C7GTH0 10820691 Ki = 86000 nM T31514 CAWL97 10888248 IC50 > 1000000 nM T31514 C06FUY 11105683 IC50 > 1000000 nM T31514 CC4N0X 11258014 IC50 > 1000000 nM T31514 CWQ40Y 11527348 IC50 = 34 ug.mL-1 T31514 CNU90T 11600756 IC50 > 1000000 nM T31514 CB5IT4 11712948 IC50 > 100 ug.mL-1 T31514 C1JBA9 11816841 IC50 = 500000 nM T31514 CO9FE0 13880378 IC50 > 300000 nM T31514 C8K0JT 15221166 Ki = 2500 nM T31514 C1GO6Q 15389575 Ki = 2600 nM T31514 C3G9LJ 20969430 IC50 = 750 nM T31514 C4HAT6 21159751 IC50 = 67.43 ug.mL-1 T31514 COK9P5 21479008 IC50 = 10.3 nM T31514 CZ21NH 23622616 IC50 > 1000000 nM T31514 C2FA6Z 36649951 IC50 = 1630 nM T31514 C6K1LC 44225039 IC50 = 16600 nM T31514 CFM53I 44322630 IC50 = 2930 nM T31514 C9SB6W 44322665 IC50 > 300000 nM T31514 C76PYN 44322883 IC50 > 118000 nM T31514 CF15IC 44322890 IC50 = 2320 nM T31514 CYBM80 44367875 IC50 > 1000000 nM T31514 CF7H4C 44368231 IC50 > 1000000 nM T31514 C75BDZ 44368232 IC50 > 1000000 nM T31514 CS5ZN1 44368239 IC50 > 1000000 nM T31514 CN7S9Z 44566965 IC50 = 4.08 ug.mL-1 T31514 CQ3SX9 44820249 IC50 = 500 nM T31514 CNL06X 44820252 IC50 = 500000 nM T31514 CQ0Z7V 44825289 IC50 = 3260 nM T31514 C0N1QJ 44825290 IC50 = 2910 nM T31514 CWE16I 44825295 IC50 = 18820 nM T31514 C5RVG0 44825296 IC50 = 94310 nM T31514 C19JRM 44825297 IC50 = 1880 nM T31514 C4W2PN 44825298 IC50 = 14940 nM T31514 CSR9I5 44825302 IC50 = 25900 nM T31514 C19FAW 44825304 IC50 = 32610 nM T31514 CNW3Q7 44825307 IC50 = 3660 nM T31514 C6OAB4 44825308 IC50 = 12980 nM T31514 CWQ71M 44825310 IC50 = 1300 nM T31514 C7VXA4 45111959 IC50 = 55000 nM T31514 CF8C3V 45375976 IC50 > 1000000 nM T31514 CVU4K0 45375977 IC50 > 1000000 nM T31514 COG49P 45483515 IC50 > 1000000 nM T31514 CT5WL3 45483523 IC50 > 1000000 nM T31514 CLE9M0 46905180 Ki = 2900 nM T31514 CBPN14 122182011 IC50 = 81700 nM T31514 C42SQJ 122182012 IC50 = 28000 nM T31514 CAST02 122182013 IC50 > 100000 nM T31514 CW1K3T 122182014 IC50 = 2200 nM T31514 CXA6K0 122182015 IC50 > 100000 nM T31514 CW67PI 122182016 IC50 = 14400 nM T31514 CH2JS1 136016326 Ki = 4000000 nM T31514 CHB13I 136016327 Ki = 700000 nM T31514 CIP40B 136056120 Ki = 5000 nM T31514 CFEO72 136056121 Ki = 100000 nM T31514 CDT8H7 137631949 IC50 = 14450 nM T31514 CH9Y7D 137635410 IC50 = 18220 nM T31514 C15VKA 137637280 IC50 = 21000 nM T31514 CKG82V 137639124 IC50 = 20170 nM T31514 CI8P4M 137639399 IC50 = 16940 nM T31514 C9V0AL 137642792 IC50 = 19130 nM T31514 C1S6KV 137646940 IC50 = 27710 nM T31514 CQ28EJ 137647619 IC50 = 17020 nM T31514 CP1TQ6 137649421 IC50 = 15970 nM T31514 CKW60Q 137656532 IC50 = 15240 nM T31514 CFV6Z5 137660606 IC50 = 11630 nM T31514 C6DRH4 137660902 IC50 = 37440 nM T31514 CVUI53 137661347 IC50 = 25690 nM T31514 D00YEV 5281605 IC50 = 500000 nM T31514 D03TYC 159496 IC50 = 100 nM T31514 D07JCA 457676 IC50 = 18000 nM T31514 D07LUJ 64945 IC50 = 4.42 ug.mL-1 T31514 D08TQA 174312 IC50 = 57000 nM T31514 D0N9IX 9822159 IC50 = 400 nM T31514 D0R8TR 445612 IC50 > 1000000 nM T81850 D0L5WM 2157 IC50 = 8000 nM T81850 D0K8DI 5274428 Ki = 740 nM T81850 D02FXU 9874248 IC50 = 78 nM T81850 D03GQH 132887 IC50 = 300 nM T81850 D0O1AV 6438355 IC50 = 5 nM T81850 CNZI26 405380 IC50 = 1290 nM T81850 C0K5BH 405389 IC50 = 240 nM T81850 C2N3TH 406065 IC50 > 100000 nM T81850 CU7BC5 406073 IC50 > 100000 nM T81850 CLI12P 460619 IC50 = 26 nM T81850 C2HT3Q 460622 IC50 = 7 nM T81850 CJCQ14 460623 IC50 = 17 nM T81850 C3MKN6 460625 IC50 = 4 nM T81850 CQ52WZ 460626 IC50 = 8 nM T81850 C4LMZ5 460628 IC50 > 200 nM T81850 C98JDN 460631 IC50 > 147 nM T81850 CL90RQ 460632 IC50 > 200 nM T81850 C36IOP 460633 IC50 > 200 nM T81850 C1MY6D 460635 IC50 = 8 nM T81850 C1F2DP 460636 IC50 = 2 nM T81850 CE49QH 460638 IC50 > 200 nM T81850 C56AQZ 460639 IC50 > 200 nM T81850 C42CWQ 6474278 IC50 > 200 nM T81850 C8WRU4 6474279 IC50 = 15 nM T81850 C69SCU 9960389 IC50 = 45 nM T81850 CFP36G 10187479 IC50 = 18 nM T81850 CZ8F6U 10350609 IC50 = 23300 nM T81850 CC1E9A 10485180 IC50 = 5000 nM T81850 C5DF4U 10875294 IC50 = 18 nM T81850 CL49WQ 10907858 IC50 = 32 nM T81850 C9X1TD 10908260 IC50 = 61 nM T81850 CR46GI 10918648 IC50 = 21 nM T81850 CUD3I8 10930227 IC50 = 70 nM T81850 CUD84P 10930347 IC50 = 87 nM T81850 CV79LB 10962885 IC50 = 38 nM T81850 CG0B5F 10985256 IC50 = 93 nM T81850 CI12XL 11123636 IC50 = 223 nM T81850 C7IP5V 11124788 IC50 = 18 nM T81850 CX16SZ 11767572 IC50 = 89 nM T81850 CJH5F0 15261219 IC50 = 350 nM T81850 C6TX5D 15261220 IC50 = 290 nM T81850 C2NX1K 15261223 IC50 = 130 nM T81850 C5H3SP 15261228 IC50 = 42 nM T81850 CMYE42 15784674 IC50 = 1900 nM T81850 CPNI32 24889304 IC50 = 169 nM T81850 C0ZQ4C 25222754 IC50 = 470 nM T81850 CXZ34C 25222756 IC50 = 1100 nM T81850 CBS1N5 25222758 IC50 = 540 nM T81850 CXQ67S 25222760 IC50 = 14 nM T81850 CP1QK2 25222763 IC50 = 32 nM T81850 C8HM3R 25222852 IC50 = 20 nM T81850 C09ANG 25222855 IC50 = 790 nM T81850 CS62IB 25223964 IC50 = 72 nM T81850 C84RHW 25223965 IC50 = 1900 nM T81850 CRVX87 25223966 IC50 = 170 nM T81850 C43JAY 25224065 IC50 = 220 nM T81850 CI73HS 25224067 IC50 = 1800 nM T81850 C3IQ5D 25224069 IC50 = 1900 nM T81850 C91WBQ 25224171 IC50 = 550 nM T81850 CV90DZ 25224172 IC50 = 79 nM T81850 CP79OV 25224173 IC50 = 69 nM T81850 C0U7DR 25224283 IC50 = 69 nM T81850 CEYM30 25224284 IC50 = 180 nM T81850 CI63GP 25224286 IC50 = 20 nM T81850 CK45GN 25224287 IC50 = 4000 nM T81850 CS47MB 25224288 IC50 = 720 nM T81850 CK1M3T 44185247 Ki = 740 nM T81850 C89AZU 44185249 Ki = 530 nM T81850 CTDS49 44185309 Ki = 1100 nM T81850 C3MGU0 44185311 Ki > 30000 nM T81850 C4LVK0 44185313 Ki = 1600 nM T81850 CQW9S5 44185315 Ki = 30000 nM T81850 CRS9U1 44185317 Ki > 30000 nM T81850 CDEF89 44185318 Ki > 30000 nM T81850 C9Y4LT 44185319 Ki = 1000 nM T81850 CN1OB7 44185377 Ki = 520 nM T81850 CP6F8I 44185379 Ki = 6200 nM T81850 CH7SB5 44185381 Ki = 300 nM T81850 CZ2BF3 44185383 Ki > 30000 nM T81850 C90XEB 44185385 Ki > 30000 nM T81850 CW4QI3 44185387 Ki = 20000 nM T81850 C6O8WD 44185389 Ki > 30000 nM T81850 C9PO0Q 44185450 Ki > 30000 nM T81850 C9CKL7 44185451 Ki > 30000 nM T81850 C4W3TA 44275230 Ki = 43 nM T81850 CW7X2H 44287785 IC50 = 0.24 nM T81850 C9MES6 44298099 IC50 = 1400 nM T81850 CBL05Y 44302736 IC50 > 300 nM T81850 C3FX0J 44302754 IC50 = 660 nM T81850 C8Z3TR 44302778 IC50 = 19 nM T81850 CKF5V4 44302831 IC50 = 1.2 nM T81850 CX8WD7 44302832 IC50 = 3.2 nM T81850 CT6GD7 44302835 IC50 > 300 nM T81850 C2R6VX 44302860 IC50 = 16 nM T81850 CB5X7N 44308457 IC50 = 430 nM T81850 CKJR49 44308477 IC50 = 8000 nM T81850 CW4Y2H 44308545 IC50 = 5 nM T81850 CU7LB4 44308575 IC50 = 1200 nM T81850 CUSC36 44318857 IC50 = 5 nM T81850 CX3W4Z 44322018 IC50 = 10 nM T81850 CKD08H 44339835 IC50 = 200 nM T81850 CR1EV9 44339899 IC50 = 7 nM T81850 C6WTK2 44339909 IC50 = 14 nM T81850 CM85WC 44339920 IC50 = 208 nM T81850 CVT5Z6 44339956 IC50 = 200 nM T81850 CQ21WM 44340057 IC50 = 9 nM T81850 C21SVY 44352756 IC50 = 0.28 nM T81850 CA1G2Z 44352820 IC50 = 3.2 nM T81850 C3H1CT 44352885 IC50 = 0.96 nM T81850 CGOK59 44352892 IC50 = 0.64 nM T81850 CJ6HA8 44360535 IC50 = 28 nM T81850 CJ60GL 44360891 IC50 = 471 nM T81850 CO1X2H 44361612 IC50 = 3.9 nM T81850 C15RIN 44380959 IC50 = 7000 nM T81850 CQ84LR 44450554 IC50 > 20000 nM T81850 CNB45X 44450555 IC50 = 1.5 nM T81850 C9HTE3 44450563 IC50 = 7000 nM T81850 C2M3WY 44450564 IC50 > 20000 nM T81850 CPCQ86 44450565 IC50 = 250 nM T81850 CC1DL6 44564237 IC50 = 17 nM T81850 CL3Q0F 44564366 IC50 = 8 nM T81850 CXP9K6 44564452 IC50 = 33 nM T81850 CK3B0E 44566224 IC50 = 0.2 nM T81850 CR1Y8L 44566225 IC50 = 4 nM T81850 C92TCB 44566226 IC50 = 2 nM T81850 C38TRS 52918309 IC50 = 220 nM T81850 C4AYK7 52939111 IC50 = 0.85 nM T81850 CYE32K 52939222 IC50 = 1.3 nM T81850 C4CNA9 52939223 IC50 = 1.1 nM T81850 CI40NH 53317065 IC50 = 2100 nM T81850 CZ35MI 53317066 IC50 > 6000 nM T81850 C2ZOM6 53317099 IC50 = 2 nM T81850 CH39BD 53317112 IC50 > 600 nM T81850 C83MKB 53317113 IC50 = 13 nM T81850 C4LZ2T 53317114 IC50 > 600 nM T81850 CE7HG9 53317115 IC50 > 600 nM T81850 CV30FT 53317117 IC50 = 8.4 nM T81850 C1ON2H 53317118 IC50 > 600 nM T81850 C95XSA 53317677 IC50 = 0.45 nM T81850 C0D6NC 53317678 IC50 > 600 nM T81850 C7WCX8 53318350 IC50 = 20 nM T81850 C7Z9IM 53318351 IC50 = 2.3 nM T81850 CF8W4Y 53318352 IC50 = 1.1 nM T81850 CTO6G8 53318353 IC50 = 260 nM T81850 CUN52D 53318354 IC50 = 600 nM T81850 C96IGD 53318394 IC50 = 1.1 nM T81850 C8THZ0 53318401 IC50 = 17 nM T81850 C1IUJ9 53318402 IC50 = 190 nM T81850 CU4C8X 53318800 IC50 = 10 nM T81850 COR5A7 53319687 IC50 = 2.4 nM T81850 CXO61Q 53319688 IC50 = 3.7 nM T81850 C58WYX 53319689 IC50 = 7.9 nM T81850 C2C9LK 53319690 IC50 = 650 nM T81850 CB10OK 53319722 IC50 > 600 nM T81850 CF2HO3 53319733 IC50 > 600 nM T81850 C0LBC4 53319734 IC50 = 7 nM T81850 C2FK5H 53319735 IC50 > 600 nM T81850 CT4QE5 53320115 IC50 = 2 nM T81850 CZ93IE 53320352 IC50 > 600 nM T81850 C95OVR 53320987 IC50 = 1700 nM T81850 C2I3LU 53320988 IC50 = 280 nM T81850 CO6SR4 53320989 IC50 = 410 nM T81850 CKF08M 53321028 IC50 > 600 nM T81850 C4HL6J 53321641 IC50 = 210 nM T81850 CB4V0W 53321661 IC50 = 220 nM T81850 C31KZN 53322331 IC50 = 130 nM T81850 CUQ5S1 53322332 IC50 > 6000 nM T81850 CI1F3J 53322368 IC50 > 600 nM T81850 CZL6P4 53322369 IC50 = 1.7 nM T81850 CE7K6D 53322370 IC50 > 600 nM T81850 CZU6I8 53322371 IC50 = 2.8 nM T81850 C7FP9Z 53322372 IC50 = 290 nM T81850 CVP2F8 53322912 IC50 = 6500 nM T81850 C4WY0P 53323688 IC50 = 21000 nM T81850 CIU4H3 53323719 IC50 = 410 nM T81850 CXG73O 53323729 IC50 = 1.3 nM T81850 CRNU30 53324348 IC50 = 97 nM T81850 CLNS96 53324963 IC50 = 770 nM T81850 C15FUS 53324994 IC50 = 7.2 nM T81850 C7XQ4R 53325006 IC50 > 600 nM T81850 C7O3XE 53325007 IC50 = 6.8 nM T81850 C6LGR3 53326264 IC50 = 1.3 nM T81850 CV8BT9 53326265 IC50 = 1.6 nM T81850 CMJF34 53326284 IC50 = 28 nM T81850 COA5G8 53326299 IC50 = 2.6 nM T81850 CSQE53 53326300 IC50 = 1700 nM T81850 C6VWB4 53326301 IC50 > 600 nM T81850 CT0E3P 53354784 IC50 = 112 nM T81850 CX0LR3 54580309 IC50 = 15300 nM T81850 CWQX70 54581312 IC50 = 2200 nM T81850 C49UFG 54581313 IC50 = 1200 nM T81850 C30EDL 54581314 IC50 = 500 nM T81850 C2K3YW 54581628 IC50 = 1420 nM T81850 CK23DS 54582322 IC50 > 20000 nM T81850 CXJF34 54582323 IC50 > 20000 nM T81850 CZN0B1 54582324 IC50 = 1900 nM T81850 CW4CP7 54582325 IC50 = 1400 nM T81850 C6U3HQ 54582326 IC50 = 370 nM T81850 CE4A7P 54582327 IC50 > 20000 nM T81850 C90GIS 54582703 IC50 = 131 nM T81850 CYG1S3 54583685 IC50 = 56 nM T81850 CP8TS5 54584271 IC50 > 20000 nM T81850 CO2B8J 54584272 IC50 = 450 nM T81850 CW9Y7D 54585229 IC50 > 20000 nM T81850 C6Q4HI 54585230 IC50 > 20000 nM T81850 CK25QX 54585231 IC50 > 20000 nM T81850 CT8VF5 54585587 IC50 = 162 nM T81850 C7J3OG 54587202 IC50 = 3300 nM T81850 CG38XD 54587203 IC50 = 5500 nM T81850 CCW8Z4 54587204 IC50 = 2400 nM T81850 C8XAD0 54587205 IC50 = 930 nM T81850 C98QBG 71452787 IC50 = 0.73 nM T81850 C30YFL 90655951 IC50 = 100000 nM T81850 CRJQ08 90655952 IC50 = 100000 nM T81850 D00KMC 56947050 IC50 = 2 nM T81850 D00YIS 56947013 IC50 = 3700 nM T81850 D01UKV 23653492 IC50 = 250 nM T81850 D03CUH 44352782 IC50 = 0.3 nM T81850 D04GSN 11814656 IC50 = 0.3 nM T81850 D06AJN 56947056 IC50 = 1 nM T81850 D06VOJ 10460101 IC50 = 0.52 nM T81850 D07ICD 11082054 IC50 = 15 nM T81850 D09ATQ 56947058 IC50 = 11700 nM T81850 D0AP5M 56947011 IC50 = 3 nM T81850 D0E1BR 56947048 IC50 = 4 nM T81850 D0G9LW 56947054 IC50 = 5 nM T81850 D0I3TX 9848748 IC50 = 2.5 nM T81850 D0NL2L 11550718 IC50 = 2800 nM T81850 D0PP5M 16730264 IC50 = 23 nM T81850 D0Q3DY 11071684 IC50 = 15 nM T81850 D0U0NT 9844255 IC50 = 6 nM T81850 D0WG7H 56947052 IC50 = 3 nM T81850 D0Z5BQ 44584870 IC50 = 660 nM T92494 D03HUX 49792852 IC50 > 10000 nM T92494 D0O0LS 25141092 IC50 > 10000 nM T92494 CNP3M1 403661 IC50 = 3200 nM T92494 CW12OJ 913113 IC50 = 220 nM T92494 C1YR8G 930898 IC50 = 2500 nM T92494 CJ5R3T 2862632 IC50 > 50000 nM T92494 C0G6HE 2887580 IC50 = 31200 nM T92494 C6C7KS 3118792 IC50 > 50000 nM T92494 C5W2KH 3934840 IC50 = 31600 nM T92494 C57YKP 4549587 IC50 > 50000 nM T92494 CMX30O 4918451 IC50 = 23800 nM T92494 CA7ZB5 5073419 IC50 = 1100 nM T92494 CP47OJ 5294673 IC50 = 47900 nM T92494 C61JMS 6419746 IC50 = 440 nM T92494 C34IZE 13381774 IC50 > 25000 nM T92494 C0PDQ8 14998467 IC50 > 25000 nM T92494 CJQ87T 14998469 IC50 > 25000 nM T92494 C2V6KL 14998470 IC50 = 420 nM T92494 C9SK0O 16771286 IC50 > 50000 nM T92494 C0BDC3 16772264 IC50 = 35100 nM T92494 CI6S4W 16772580 IC50 = 29300 nM T92494 CTH5M9 24696534 IC50 > 50000 nM T92494 CU3RF1 45139989 IC50 > 10000 nM T92494 CQGZ06 45139991 IC50 > 10000 nM T92494 CRF27I 45439084 IC50 = 37800 nM T92494 CL3YZ6 45439117 IC50 > 50000 nM T92494 CLOY23 45439122 IC50 = 18700 nM T92494 C9SNG3 45439130 IC50 > 50000 nM T92494 CPY1V7 45439136 IC50 = 19600 nM T92494 C7ON5A 46233287 IC50 > 10000 nM T92494 CU07GH 46830215 IC50 = 170 nM T92494 C8LUR2 46830216 IC50 = 320 nM T92494 CF79OC 46884078 IC50 = 1100 nM T92494 C3XDZ1 46884079 IC50 = 860 nM T92494 CV5F1S 46884080 IC50 = 2000 nM T92494 CDZJ97 46884081 IC50 = 10000 nM T92494 C6O7NM 46884082 IC50 = 990 nM T92494 C1ITW4 46884083 IC50 = 1100 nM T92494 C2YHB9 46884124 IC50 > 20000 nM T92494 CY9CM0 46884125 IC50 = 860 nM T92494 CE16JN 46884126 IC50 = 1300 nM T92494 C3U6AF 46884127 IC50 = 1200 nM T92494 C59XDL 46884128 IC50 = 640 nM T92494 C2VEK3 46884159 IC50 = 460 nM T92494 CVU2S1 46884160 IC50 = 940 nM T92494 C0DVM6 46884161 IC50 = 990 nM T92494 CV0CZ2 46884162 IC50 = 1100 nM T92494 C3JUP8 46884205 IC50 = 1400 nM T92494 CJCY89 46884206 IC50 > 20000 nM T92494 C0ONT9 46884207 IC50 > 20000 nM T92494 CR3E9J 46884208 IC50 = 280 nM T92494 C2GD3A 46884209 IC50 = 300 nM T92494 CP7E2Q 46884244 IC50 = 330 nM T92494 CY12AZ 46884245 IC50 = 660 nM T92494 CP56VB 46884246 IC50 = 800 nM T92494 C7FM0X 46884247 IC50 = 1100 nM T92494 C3OTV6 46884248 IC50 > 20000 nM T92494 C8N2TY 46884286 IC50 > 20000 nM T92494 CZ1I9U 46884287 IC50 > 20000 nM T92494 CNQ28F 46884288 IC50 > 10000 nM T92494 C2A4KI 46884357 IC50 > 10000 nM T92494 C8F6BQ 46884358 IC50 > 10000 nM T92494 C4E1HD 46884359 IC50 = 3700 nM T92494 CIY69W 46884360 IC50 = 350 nM T92494 C6DR3V 46884361 IC50 > 20000 nM T92494 C8SB6Z 46884407 IC50 = 110 nM T92494 C48MWS 46884408 IC50 = 4700 nM T92494 CF91RS 49843531 IC50 > 10000 nM T92494 C2Y6QS 50938552 IC50 > 10000 nM T92494 C9NYP4 51036677 IC50 > 10000 nM T92494 C4WRY3 51037112 IC50 > 10000 nM T92494 CRI28Z 51037948 IC50 > 10000 nM T92494 CCN01X 71547862 IC50 > 10000 nM T92494 CY0UC4 90645194 IC50 > 10000 nM T92494 CY7BI2 118706214 IC50 > 10000 nM T92494 CRT04G 118711588 IC50 = 1000 nM T92494 CU4M9B 118711589 IC50 > 25000 nM T92494 CXMK27 118711590 IC50 > 25000 nM T92494 CJU0E4 118712153 IC50 = 6600 nM T92494 CKN5Z0 118712155 IC50 = 930 nM T92494 C0LZX3 118712156 IC50 > 25000 nM T92494 C1FB0H 118712157 IC50 > 25000 nM T92494 C21ZVJ 118712158 IC50 > 25000 nM T92494 CHA4N2 136013680 IC50 > 10 nM T92494 C1YUD0 136219394 IC50 > 10 nM T92494 CIU8W3 136254389 IC50 > 10 nM T92494 C80OCM 145949854 IC50 = 60 nM T92494 CL2K0H 145950254 IC50 = 17100 nM T92494 CC45BE 145950371 IC50 = 28400 nM T92494 C6E2QW 145950757 IC50 = 12500 nM T92494 CKM97I 145950826 IC50 = 11600 nM T92494 CVU03H 145951159 IC50 > 50000 nM T92494 C3DYT1 145952180 IC50 = 33700 nM T92494 CINV23 145952466 IC50 = 38500 nM T92494 CRK2O7 145952677 IC50 = 27500 nM T92494 C2YI1P 145953283 IC50 > 50000 nM T92494 CXLQ63 145953404 IC50 > 50000 nM T92494 CT7K6J 145953445 IC50 = 33400 nM T92494 C1JL6H 145954134 IC50 > 50000 nM T92494 CTN1O4 145954990 IC50 > 50000 nM T92494 C92OAW 145955902 IC50 = 44500 nM T92494 C31SEA 145956246 IC50 = 19900 nM T92494 CXFR20 145956929 IC50 > 50000 nM T92494 C16RDC 145957256 IC50 = 22600 nM T92494 C9DSA0 145957433 IC50 = 36700 nM T92494 CR42VN 145958351 IC50 > 50000 nM T92494 CW8J1R 145958740 IC50 > 50000 nM T92494 CAZ85N 145958943 IC50 = 5500 nM T92494 CY8S1O 145959480 IC50 = 44400 nM T92494 CMDH42 145959604 IC50 = 11700 nM T92494 CBJ9C3 145959921 IC50 > 50000 nM T92494 C0BWK5 145959938 IC50 > 50000 nM T92494 CRKD16 145959989 IC50 = 19400 nM T92494 C3OHS2 145962282 IC50 = 44500 nM T92494 CLPT25 145963535 IC50 = 18400 nM T92494 CC38RD 145971446 IC50 > 50000 nM T92494 C0J7KQ 145974054 IC50 = 9500 nM T92494 CWL50V 145981755 IC50 = 762 nM T92494 C2MD1Q 155513187 IC50 > 10000 nM T92494 D08HFG 24809764 IC50 > 10000 nM T92494 D09HVH 135566652 IC50 > 10 nM T99908 CKO4M6 56663319 Ki = 68 nM T99908 CY34VE 56677007 Ki = 53 nM T99908 D07ZRG 46899577 Ki = 20 nM T77796 D0E9TD 638678 EC50 = 3 nM T77796 CSJB84 16066773 Ki = 3.2 nM T77796 CO3S8K 44422085 Ki > 100000 nM T77796 CCL53X 44422086 Ki > 100000 nM T77796 CSG40O 44422091 EC50 > 100000 nM T77796 CL3B5P 44422092 Ki > 100000 nM T77796 CB1U5O 44422097 Ki > 100000 nM T77796 CA1C8X 44422098 Ki > 100000 nM T77796 CW1Q5S 44422105 Ki > 100000 nM T77796 CHL12A 44422106 Ki > 100000 nM T77796 C5RLY3 44422110 Ki > 100000 nM T77796 CI7D8W 44422111 Ki > 100000 nM T77796 CNI83Z 44422115 Ki > 100000 nM T77796 CTO4Y3 44422122 Ki = 3 nM T77796 C37EAR 44422168 Ki = 11 nM T77796 CGJ71P 44422169 EC50 = 17000 nM T77796 COGC73 44422176 EC50 = 5100 nM T77796 CU8WO6 44422177 EC50 = 380 nM T84780 D01NUR 118169620 IC50 = 0.22 nM T84780 D03MXK 25022340 Ki = 1.9 nM T84780 D07CLV 46940575 IC50 = 10.4 nM T84780 D09MIN 24737642 EC50 = 0.4 nM T84780 D0E8NP 49836020 IC50 = 50 nM T84780 D0Q7AG 53240420 IC50 > 50000 nM T84780 D08UPQ 73603510 IC50 = 7 nM T84780 D0YN1X 71661892 Ki = 3.7 nM T84780 CE1Q0I 7019981 IC50 = 24000 nM T84780 CO1ZE4 9927170 IC50 = 690 nM T84780 C2IAF0 10222526 IC50 = 0.32 nM T84780 CWZ8F7 11503417 IC50 = 27 nM T84780 CY3RV2 17756618 Ki = 0.5 nM T84780 CBM94F 23646361 Ki = 188 nM T84780 C8XJG1 24754961 Ki > 3000 nM T84780 C0X8NI 24939290 IC50 = 530 nM T84780 C7XTN2 25138055 Ki = 3 nM T84780 CJ2VZ4 25138056 Ki = 1.1 nM T84780 C29PBM 25138057 Ki = 150 nM T84780 CLO6Y8 25138058 Ki = 13 nM T84780 CPN8E5 25138069 Ki = 0.68 nM T84780 CWH17B 25138070 Ki = 29 nM T84780 C0BJQ6 25173661 Ki = 7300 nM T84780 CSD59K 25173742 Ki = 1.2 nM T84780 C8DZE7 25180121 Ki = 3.3 nM T84780 CY0A9T 25180312 Ki = 3.7 nM T84780 CW4U0R 25180313 Ki = 1.1 nM T84780 C2SWF7 25195345 Ki = 129 nM T84780 C46SKW 25195346 Ki = 33 nM T84780 CAL8M3 25209021 Ki = 0.37 nM T84780 CD29TU 25209022 Ki = 1.27 nM T84780 CU07LB 44237069 IC50 = 1.42 nM T84780 CDW4O5 44567555 IC50 = 1060 nM T84780 C2JT3G 44567559 IC50 = 12100 nM T84780 CB5A3P 44567560 IC50 = 24100 nM T84780 CQ48DW 44567561 IC50 = 45200 nM T84780 C0X6IF 44567562 IC50 = 19900 nM T84780 C0TMS1 44567563 IC50 = 1540 nM T84780 C5N1FL 44567564 IC50 = 1250 nM T84780 CD4B1V 44567568 IC50 > 20000 nM T84780 C6WPZ4 44567569 IC50 = 840 nM T84780 C8QO7F 44567571 IC50 = 4690 nM T84780 C12NPW 44567572 IC50 = 9200 nM T84780 CO8G3P 44596256 IC50 < 2 nM T84780 C96OTK 46830178 Ki = 11 nM T84780 CECL56 46830179 Ki = 161 nM T84780 C8RDC3 46888403 Ki = 84 nM T84780 CP40QG 46929436 Ki = 1.6 nM T84780 CQ0A5I 46929438 Ki = 12.2 nM T84780 C5FK8W 46929440 Ki < 1 nM T84780 C1TIK8 46930628 Ki = 7.9 nM T84780 CVC3T5 46930723 Ki = 6.6 nM T84780 CK4R2U 49800198 EC50 = 0.2 nM T84780 CUG1X6 49847567 EC50 = 0.1 nM T84780 CD1G0B 50913340 IC50 = 2.1 nM T84780 CNQO70 52951104 Ki < 1 nM T84780 C30GIF 53237922 Ki = 2 nM T84780 CW7AF2 53238154 Ki = 1 nM T84780 C5JPH2 53238155 Ki = 1 nM T84780 CW71DY 53238387 Ki = 1 nM T84780 C16JNG 53238388 Ki = 2 nM T84780 C3IPJ4 53238615 Ki < 1 nM T84780 CH0L8C 53238616 Ki < 1 nM T84780 CF83PC 53238842 Ki = 1 nM T84780 C2HB0C 53238843 Ki = 1 nM T84780 C7SR2W 53239063 Ki < 1 nM T84780 CM46PV 53239064 Ki = 1 nM T84780 CNFD80 53239285 Ki = 2 nM T84780 CCL6I5 53239286 Ki = 3 nM T84780 C61NHL 56945169 Ki = 1.2 nM T84780 C2WXP5 56945170 Ki = 2 nM T84780 C7YW1J 56945269 Ki = 1.9 nM T84780 CR7TD9 56945270 Ki = 2.9 nM T84780 CAD3P5 56945392 Ki = 1.2 nM T84780 CDYL09 56945393 Ki = 3.6 nM T84780 C7X1ZF 56946798 Ki = 0.7 nM T84780 C05JAE 56946799 Ki = 0.4 nM T84780 C8IWF7 57345674 IC50 < 2 nM T84780 COLI80 57390699 EC50 = 300 nM T84780 CMCA76 57390756 EC50 = 185 nM T84780 CY1AO9 57390796 IC50 = 1690 nM T84780 CH9Z4T 57390797 IC50 = 270 nM T84780 CO9N3Z 57391385 IC50 < 2 nM T84780 CIP23W 57391386 IC50 < 2 nM T84780 C9FIB5 57391387 IC50 = 2.6 nM T84780 CAU17J 57392501 IC50 = 62 nM T84780 C8W3UM 57392502 IC50 = 33 nM T84780 CB9HN3 57392503 IC50 = 301 nM T84780 CJ94CH 57392610 IC50 = 740 nM T84780 C1W8YU 57392611 IC50 = 790 nM T84780 C6QHW5 57393149 IC50 < 2 nM T84780 CLJ61G 57394210 IC50 = 5750 nM T84780 CKXM93 57394211 IC50 = 18 nM T84780 C6SN2U 57394212 IC50 = 24 nM T84780 CQHV21 57394330 IC50 = 130 nM T84780 CO84WG 57395973 IC50 = 26 nM T84780 C2AR4B 57395974 IC50 = 44 nM T84780 CUG3R7 57395975 EC50 = 279 nM T84780 CH1X6S 57395976 IC50 = 52 nM T84780 CQ1IW8 57395977 EC50 = 158 nM T84780 CN0AF2 57396041 IC50 = 4 nM T84780 CLU86I 57396085 IC50 = 5020 nM T84780 CUB1H9 57396086 IC50 = 740 nM T84780 CXS64P 57396647 IC50 < 2 nM T84780 CP2FN7 57397775 IC50 = 3890 nM T84780 CF3LE6 57397776 EC50 = 156 nM T84780 CH98VA 57397777 IC50 = 24 nM T84780 CT0AE9 57397898 IC50 = 500 nM T84780 CD0O6B 57397899 IC50 = 780 nM T84780 C9G7YF 57398349 IC50 < 2 nM T84780 CS40ZQ 57399437 IC50 = 1990 nM T84780 C1KRZ0 57399438 IC50 = 30 nM T84780 C8WZ1A 57400074 IC50 < 2 nM T84780 CHD41O 57400075 IC50 < 2 nM T84780 CG4B9T 57400076 IC50 < 2 nM T84780 C5N4FG 57400077 IC50 < 2 nM T84780 C9Q5WO 57400078 IC50 < 2 nM T84780 C6ZY0D 57400338 EC50 = 113 nM T84780 C1D5OW 57401193 IC50 = 80 nM T84780 C6IT0P 57401194 IC50 = 20 nM T84780 CGC3F0 57401195 EC50 = 68 nM T84780 CFU7D8 57401196 EC50 = 60 nM T84780 CZ2K9F 57401197 IC50 = 593 nM T84780 CR06YF 57401295 IC50 = 3380 nM T84780 C2FKB1 57401296 IC50 = 3360 nM T84780 C5DK7R 57401297 IC50 = 450 nM T84780 C9IB0C 57401812 IC50 < 2 nM T84780 CZP8Q6 57401885 IC50 < 2 nM T84780 C9CRY4 57401886 IC50 < 2 nM T84780 CKU4F8 57403521 IC50 < 2 nM T84780 CESB84 57403599 IC50 = 3.3 nM T84780 CE6SU4 57689264 Ki < 0.5 nM T84780 C62ZCQ 57689338 Ki = 13.7 nM T84780 CF89OA 58137904 IC50 = 2.2 nM T84780 C3KDR0 58609608 IC50 = 48.2 nM T84780 C1C7ML 59542215 IC50 <= 1 nM T84780 CJL17T 60198193 IC50 = 1 nM T84780 C3QS0C 60198300 IC50 = 1.1 nM T84780 C16DYA 60198985 IC50 = 1.4 nM T84780 CW9U7M 66972432 IC50 = 1.2 nM T84780 C06KWB 66972973 IC50 = 3.5 nM T84780 C0VG8C 66973046 IC50 = 28 nM T84780 CQ1O6Z 66973400 IC50 = 2.1 nM T84780 COQ52M 70678411 IC50 = 5.4 nM T84780 CM65DI 70980530 EC50 = 0.32 nM T84780 CO8YK2 70981017 IC50 = 10 nM T84780 C63JLP 71450435 IC50 = 1.4 nM T84780 C9BCY8 71452258 IC50 <= 1 nM T84780 CL31QP 71452260 IC50 = 3.2 nM T84780 C9QF2G 71452262 IC50 = 1.4 nM T84780 CCGT91 71452264 IC50 = 1.7 nM T84780 CS4V9B 71452266 IC50 = 3.8 nM T84780 CM14JU 71454062 IC50 = 1.5 nM T84780 CL3KX5 71454063 IC50 = 12.6 nM T84780 CQ8R3E 71454065 IC50 = 3.5 nM T84780 CZR6J5 71454067 IC50 <= 1 nM T84780 C4JXM9 71454115 IC50 = 17.6 nM T84780 C90KFN 71457579 IC50 = 1.7 nM T84780 CG8X3Z 71457581 IC50 = 2.9 nM T84780 C82EPD 71457647 IC50 = 2.6 nM T84780 C24OXD 71459481 IC50 = 5 nM T84780 CTV86H 71459483 IC50 <= 1 nM T84780 CMKI17 71459485 IC50 = 1.9 nM T84780 CCS3R8 71461288 IC50 = 1.5 nM T84780 CSGH36 71463006 IC50 = 1.1 nM T84780 C5HTZ1 71472009 IC50 = 3700 nM T84780 CEH3B5 71472080 IC50 = 20000 nM T84780 C7QZX1 71472243 IC50 = 650 nM T84780 C1NV7Q 71528757 EC50 = 6700 nM T84780 CY83OB 71571046 EC50 = 1400 nM T84780 CVPJ20 71581702 EC50 = 70 nM T84780 CP9G3R 71581703 EC50 = 45 nM T84780 C3F4OT 71581838 EC50 = 59 nM T84780 CLIU93 71582189 EC50 = 30 nM T84780 C1VME6 71582339 IC50 = 3 nM T84780 CZ8DF4 71661893 Ki = 7.4 nM T84780 CB0O2T 71662077 Ki = 4.7 nM T84780 COCI81 71662078 Ki = 4.9 nM T84780 CNU16X 71662256 Ki = 1.5 nM T84780 CJRL34 71662257 Ki = 5.4 nM T84780 C2UM5A 71662420 Ki = 5.8 nM T84780 CVZK59 71662421 Ki = 3.9 nM T84780 CW4G0O 71662584 Ki = 8.7 nM T84780 C8AY6G 71662585 Ki = 5 nM T84780 C3DAU6 72704974 IC50 = 4.9 nM T84780 C1B7OJ 72704975 IC50 = 3.6 nM T84780 CE1LT4 72705161 IC50 = 2.9 nM T84780 CE6J7U 72705162 IC50 = 4.5 nM T84780 CE37QK 72713171 IC50 = 271 nM T84780 C7SZ3V 72714058 IC50 = 2640 nM T84780 C5RD2F 72736709 IC50 = 1.4 nM T84780 CEK93U 72736862 IC50 = 2.8 nM T84780 C47KWN 72736863 IC50 = 1.7 nM T84780 CLMK36 73505797 IC50 = 4 nM T84780 CBK19E 73505798 IC50 = 4.8 nM T84780 CNAY12 73506219 IC50 = 10 nM T84780 CL35VQ 73506880 IC50 = 5.6 nM T84780 CJG8B6 73507094 IC50 = 4.7 nM T84780 C8QPX7 73507318 IC50 = 2 nM T84780 CKS45Y 73508005 IC50 = 0.19 nM T84780 C4K3BG 73508016 IC50 = 0.17 nM T84780 CETB68 73603641 IC50 = 5 nM T84780 C1A9ME 73672184 IC50 = 1.6 nM T84780 CJ38WP 73672428 IC50 = 0.2 nM T84780 CVOY02 73672545 IC50 = 1 nM T84780 CN3A1V 73672620 IC50 = 3.5 nM T84780 CALJ56 73672900 IC50 = 3.8 nM T84780 C8T2AC 73672902 IC50 = 0.34 nM T84780 C76XRT 73673026 IC50 = 1.3 nM T84780 CX95NQ 73673152 IC50 = 6.5 nM T84780 CPVS10 73673158 IC50 = 0.74 nM T84780 CF9GW8 73673640 IC50 = 2.5 nM T84780 CZR15M 76310221 EC50 > 370 nM T84780 C79CEF 76310225 EC50 = 0.2 nM T84780 CHG1M7 76310226 EC50 = 0.2 nM T84780 CI65XY 76310227 EC50 = 0.6 nM T84780 CVD7A2 76313911 EC50 = 5 nM T84780 CP34JE 76317444 EC50 = 0.6 nM T84780 C1VUI3 76317445 EC50 = 124 nM T84780 C7L6XM 76317446 EC50 = 15 nM T84780 C87QOG 76317450 IC50 = 290 nM T84780 C3UVM9 76321179 EC50 = 0.6 nM T84780 CG5F9W 76321180 EC50 = 4 nM T84780 C7VPM6 76324806 EC50 = 0.2 nM T84780 C31BXK 76324810 EC50 = 4 nM T84780 CW3D4U 76328360 EC50 = 3 nM T84780 CJY31H 76328361 EC50 > 370 nM T84780 CA14LJ 76328363 EC50 = 10 nM T84780 C4G8MQ 76332032 EC50 = 0.1 nM T84780 CH8I6K 76332036 EC50 > 370 nM T84780 C3VHF8 76335638 EC50 = 2 nM T84780 CMU7C4 76335639 EC50 > 370 nM T84780 CUA9F5 76335643 EC50 = 0.5 nM T84780 CQOA73 76335644 EC50 = 0.3 nM T84780 CJ9A3T 76335645 IC50 = 40 nM T84780 CR6T9Q 76335646 EC50 = 2 nM T84780 C2UVF7 76335647 EC50 = 0.1 nM T84780 CX0R6S 86276147 IC50 = 3 nM T84780 C9PHL5 89569624 IC50 = 7 nM T84780 CBL23Q 90089551 IC50 = 17 nM T84780 CBOP84 90089572 IC50 = 79 nM T84780 C73MBT 90089727 IC50 = 76 nM T84780 CO96QE 90089737 IC50 = 25 nM T84780 C10KBD 90231909 IC50 = 14 nM T84780 C3JK9T 90231969 EC50 = 150 nM T84780 CW98BE 90232119 EC50 = 20 nM T84780 CE6W1R 90232149 EC50 = 2.5 nM T84780 C75QBJ 90232154 EC50 = 7.5 nM T84780 C35JLR 90232165 EC50 = 24 nM T84780 CDP7U6 90232174 EC50 = 2.4 nM T84780 CN4D0A 90232202 EC50 = 2.3 nM T84780 CW74HX 90232234 EC50 = 240 nM T84780 C8IQ1M 90232300 EC50 = 2.4 nM T84780 C7XF3W 90251750 IC50 = 320 nM T84780 CMU3A7 90654375 IC50 = 100 nM T84780 CJQ78L 90654376 IC50 = 73 nM T84780 C6CMZ9 90654377 IC50 = 37 nM T84780 CY56XM 90654378 IC50 = 42 nM T84780 CHC78P 90654379 IC50 = 44 nM T84780 CTHF31 90654380 IC50 = 89 nM T84780 C6K0WI 90654381 IC50 = 180 nM T84780 C3HEA9 90654382 IC50 = 63 nM T84780 CA9HX4 90654383 IC50 = 290 nM T84780 CN6M3I 90654384 IC50 = 400 nM T84780 C9K0OL 90654385 IC50 = 1900 nM T84780 CORF34 90654386 IC50 = 2500 nM T84780 CO21FQ 90654387 IC50 = 450 nM T84780 CP85YF 90654388 IC50 = 1300 nM T84780 CHMQ92 90654389 IC50 = 320 nM T84780 C72LMU 90654390 IC50 = 510 nM T84780 CSE3L7 90654391 IC50 = 2800 nM T84780 CJ3Z7O 90654392 IC50 = 9500 nM T84780 CZSK32 90654393 IC50 = 1200 nM T84780 CYM9Z1 90654394 IC50 = 66 nM T84780 COTH12 90654395 IC50 = 370 nM T84780 CG5XS4 90654396 IC50 = 940 nM T84780 C7GJS1 90654397 IC50 > 10000 nM T84780 C6NW4S 90654398 IC50 = 220 nM T84780 C6YW1O 90654399 IC50 = 52 nM T84780 CN0V9Q 90654400 IC50 = 220 nM T84780 C5JLE7 90654401 IC50 = 2800 nM T84780 COR48A 90654402 IC50 = 8000 nM T84780 CIZQ28 90654403 IC50 = 50 nM T84780 CI9Q7H 90654404 IC50 = 39 nM T84780 CSB8J0 90654405 IC50 = 24 nM T84780 CCQ73R 90654406 IC50 = 35 nM T84780 CD46OI 90654407 IC50 = 21 nM T84780 CI23DO 90654408 IC50 = 44 nM T84780 C1A9HP 90654409 IC50 = 70 nM T84780 C10DYO 90654410 IC50 = 160 nM T84780 CM6S3P 90654411 IC50 = 55 nM T84780 CM59ZC 90654412 IC50 = 36 nM T84780 CZNT70 90654413 IC50 > 10000 nM T84780 CI3MX1 91826683 IC50 = 27000 nM T84780 C19PJK 91826688 IC50 = 410000 nM T84780 CF6GT5 117710478 IC50 = 3.4 nM T84780 CA67UG 118323269 IC50 = 25 nM T84780 CGH23J 118497874 IC50 = 3.4 nM T84780 C0DGE4 118497975 IC50 = 11 nM T84780 C9BSI6 118557690 IC50 = 4.2 nM T84780 CY82JZ 118557732 IC50 = 0.62 nM T84780 C6VWZ8 118557745 IC50 = 2.3 nM T84780 CH42OT 118715865 IC50 = 8 nM T84780 CHS36B 118732584 IC50 = 4.2 nM T84780 CI69WD 118732795 EC50 = 34 nM T84780 CT3OK0 126502413 IC50 = 0.13 nM T84780 C6G3QT 126502414 IC50 = 0.1 nM T84780 C0QVU3 126502417 IC50 = 0.18 nM T84780 COM04R 126502421 IC50 = 0.7 nM T84780 C6NFD0 134419123 IC50 = 220 nM T84780 CJVY85 137639402 IC50 = 1.35 nM T84780 CE1O5K 137642617 IC50 = 1.52 nM T84780 C2D3UZ 137651764 IC50 = 6.08 nM T84780 CN9C2F 137658721 IC50 = 1.66 nM T84780 CK0IX4 137662073 IC50 = 1.09 nM T84780 C87BOG 138377561 IC50 = 4.8 nM T84780 C0B8GK 138377594 IC50 = 86 nM T84780 CA43ML 142585287 IC50 > 1000 nM T84780 CGF6R2 142585309 IC50 > 1000 nM T84780 C0HC8R 142585337 IC50 = 352.6 nM T84780 C0RHF1 142585361 IC50 > 16000 nM T84780 C5AI8Z 142585365 IC50 > 5000 nM T84780 CM7IG2 142585375 IC50 > 2000 nM T84780 CG46IU 145954838 IC50 > 1000 nM T84780 CZ25IO 145957358 IC50 = 0.59 nM T84780 CKEJ30 145979040 IC50 > 200 nM T84780 C7XM4Q 145979112 IC50 = 23.9 nM T84780 CLRM52 145979809 IC50 = 181 nM T84780 CGN1J0 145980475 IC50 = 143.5 nM T84780 CL4F9B 145981512 IC50 = 1203 nM T84780 C1K6AY 145982930 IC50 > 1000 nM T84780 C3L1ZW 145985393 IC50 = 17.2 nM T84780 CY8JR0 145986444 IC50 = 197.6 nM T84780 C1HWA3 145988725 IC50 = 264.1 nM T84780 CX7AV2 145991404 IC50 = 21.7 nM T84780 C79EXP 145992527 IC50 = 4.5 nM T84780 CK8JB2 155512591 IC50 = 20 nM T84780 CEH0W4 155523271 IC50 > 200 nM T84780 C23UZA 155554597 IC50 = 15 nM T84780 CR3UQ4 155561157 IC50 = 14 nM T84780 D03KZH 25172871 Ki = 1.3 nM T84780 D0BW7P 44589292 Ki = 1.3 nM T84780 D0Q7TL 24754886 Ki = 0.8 nM T84780 D0VK7M 49847690 EC50 = 0.1 nM T50942 CCE6F2 2826530 IC50 = 3720 nM T50942 CWT83F 9885305 IC50 = 200 nM T50942 C0UN8P 9970195 IC50 = 2300 nM T50942 CX38UT 11820221 IC50 = 3100 nM T50942 CXLW54 11948707 Ki > 10000 nM T50942 CK7J6D 17756791 IC50 = 244000 nM T50942 CNM23H 44358481 IC50 = 1300 nM T50942 CP9TR0 10324985 Ki > 10000 nM T87109 D05ADP 160355 IC50 = 10000 nM T87109 D03BNU 59604787 IC50 > 10000 nM T87109 D00OWF 5280953 IC50 = 1500 nM T87109 D0F8DL 176155 IC50 = 120 nM T87109 CB1VW3 1400 IC50 = 170 nM T87109 CEC30Q 3674 IC50 = 1000 nM T87109 CJ17AM 4877 IC50 = 150 nM T87109 CBPM40 4878 IC50 = 41 nM T87109 CN64JR 8323 IC50 = 660 nM T87109 C3W0FN 591403 IC50 = 330 nM T87109 C3J1EO 591698 IC50 = 2500 nM T87109 CDM7S2 670752 IC50 = 2220 nM T87109 CVO75W 670753 IC50 = 290 nM T87109 CG3L0P 708592 IC50 = 750 nM T87109 C4U7XJ 750458 IC50 = 1090 nM T87109 C0B4AI 770971 IC50 = 570 nM T87109 CG3OU2 830481 IC50 = 1960 nM T87109 CI6X4A 886576 IC50 = 1110 nM T87109 CCU3D7 1147778 IC50 = 2690 nM T87109 CZT40M 1360240 IC50 = 2820 nM T87109 CIR4L3 1407374 IC50 = 3580 nM T87109 CAV19R 2360773 IC50 > 10000 nM T87109 C2ZU8B 2549232 IC50 = 3430 nM T87109 CV9Q7F 2596899 IC50 = 9710 nM T87109 CVIC03 2596990 IC50 = 1120 nM T87109 C3RD9H 2596997 IC50 = 1240 nM T87109 C0K9MA 2597029 IC50 = 420 nM T87109 CQU0E5 2641094 IC50 = 1170 nM T87109 CW5Y1L 2677056 IC50 = 17430 nM T87109 CT1UL5 2677057 IC50 = 5760 nM T87109 CZVN70 2677091 IC50 = 990 nM T87109 CR2ZU0 3570197 IC50 = 1430 nM T87109 CPQV76 5353678 IC50 = 700 nM T87109 CEV4X1 7719944 IC50 = 320 nM T87109 CYA76E 9798589 IC50 > 100000 nM T87109 CEW4U6 10021535 IC50 = 848 nM T87109 CBOP58 11293798 Ki > 10000 nM T87109 C26BZX 11362471 Ki > 10000 nM T87109 CWXB93 11397177 Ki > 10000 nM T87109 CXBU49 11502255 IC50 = 1400 nM T87109 CTG83F 11539329 Ki > 7800 nM T87109 CMIL86 11590363 Ki > 7800 nM T87109 C9T6SC 11640926 Ki > 7800 nM T87109 C7T9ES 11681588 IC50 = 7.8 nM T87109 C1EUQ4 12211285 IC50 = 7290 nM T87109 CFPW41 16007116 Ki > 7800 nM T87109 CZL8G5 16115351 IC50 = 230 nM T87109 CDWC87 17168177 IC50 = 260 nM T87109 CB4JP2 17395533 IC50 = 6330 nM T87109 CEX4S6 20789070 IC50 = 134 nM T87109 CJ76FL 22037373 IC50 = 545 nM T87109 C2P0VU 24247294 IC50 = 620 nM T87109 CY8L7E 24896769 IC50 > 10000 nM T87109 C5Y6GM 24901423 IC50 = 700 nM T87109 CLZ23U 24951610 IC50 > 30000 nM T87109 C2KY1G 25094210 IC50 = 1900 nM T87109 C6BWZ8 25145145 IC50 > 100 nM T87109 C78YWA 25145716 IC50 > 500 nM T87109 C6FGQ1 25206346 IC50 > 10000 nM T87109 CLW32V 27899321 IC50 = 79 nM T87109 CU9E4P 42629114 IC50 > 10000 nM T87109 CCB1E9 44124695 IC50 > 100000 nM T87109 C3VRO9 44557921 IC50 > 10000 nM T87109 CF90OX 44576212 IC50 = 400 nM T87109 C2RY3H 44597108 IC50 = 2500 nM T87109 CFD21J 44597110 IC50 = 1600 nM T87109 CS7M8K 44597113 IC50 = 110 nM T87109 CZ49BI 44597224 IC50 = 820 nM T87109 C6ET3K 44597225 IC50 = 33 nM T87109 C7D8ZN 44597226 IC50 = 4 nM T87109 C4HN5F 44597227 IC50 = 5 nM T87109 C6E2SC 45482700 IC50 > 10000 nM T87109 CZXH74 45482750 IC50 > 10000 nM T87109 CUA97D 46209401 IC50 > 10000 nM T87109 CY3HW5 46224684 IC50 = 530 nM T87109 CI1F5C 46239840 IC50 = 320 nM T87109 COTJ39 46863083 IC50 = 12000 nM T87109 CLS29B 46872626 IC50 > 10000 nM T87109 C2O8RZ 46886323 IC50 = 740 nM T87109 CBS64G 49830252 IC50 = 12000 nM T87109 C2Q0GE 50990922 IC50 = 16000 nM T87109 CAZQ43 51003133 IC50 > 1000 nM T87109 CXA03W 52920796 IC50 > 100 nM T87109 C6OTY5 53251320 IC50 > 30000 nM T87109 CE8OY2 53317913 IC50 > 100 nM T87109 C0SWH5 53348216 IC50 > 40000 nM T87109 C2EK8Z 53352108 IC50 = 83 nM T87109 CD9HS6 53352109 IC50 = 1210 nM T87109 C6O7VL 53357600 IC50 = 6.6 nM T87109 CBOD63 56835089 IC50 = 11000 nM T87109 COT01X 57382333 IC50 = 13 nM T87109 COTF12 57382553 IC50 = 42.1 nM T87109 CD6Y9Z 57395116 IC50 = 6610 nM T87109 C8W6IG 57395117 IC50 = 1730 nM T87109 CG7S0D 57396882 IC50 > 30000 nM T87109 C0UDY9 57401151 IC50 > 30000 nM T87109 CXF3R4 57411943 IC50 = 85 nM T87109 CKCR14 57411948 IC50 = 98 nM T87109 C6BPR2 58985201 IC50 > 30000 nM T87109 CT3EW2 59292007 IC50 > 1000 nM T87109 CON8H1 59326984 IC50 = 5770 nM T87109 CSRB50 60196190 IC50 = 37 nM T87109 CPU7N9 60196195 IC50 = 44 nM T87109 C7LZ5Y 60196202 IC50 = 80 nM T87109 C4PHO3 60196210 IC50 = 89 nM T87109 CK6WO0 66552478 IC50 < 10000 nM T87109 CIM7H1 66575095 IC50 = 40 nM T87109 CV63UL 67240318 IC50 > 10000 nM T87109 C1WH7K 70679288 IC50 = 22 nM T87109 CI8EG4 70682610 IC50 = 2370 nM T87109 CJ1RE5 70682611 IC50 = 1660 nM T87109 C2MPQ3 70686838 IC50 = 2620 nM T87109 CU90LB 70686839 IC50 = 4370 nM T87109 C1MCQ3 70691009 IC50 = 3170 nM T87109 CCJH52 70691010 IC50 = 2180 nM T87109 C39DER 70691011 IC50 = 2880 nM T87109 CLZ4Q1 70691012 IC50 = 3970 nM T87109 CAJF37 70693140 IC50 = 1630 nM T87109 C2U7ES 70693141 IC50 = 3610 nM T87109 CQ75AH 70693142 IC50 = 2320 nM T87109 CC48LS 70695212 IC50 = 1080 nM T87109 C56HSY 70695213 IC50 = 2180 nM T87109 CX61EW 70697244 IC50 = 3170 nM T87109 C1IEJ2 70789254 IC50 = 238000 nM T87109 C8T7ZP 70789255 IC50 = 97000 nM T87109 CH0B8N 70789756 IC50 > 30000 nM T87109 C7VA0I 71450358 IC50 = 202 nM T87109 CZ2OE6 71452173 IC50 = 68 nM T87109 CSPN93 71452174 IC50 = 15 nM T87109 CR53ZS 71452175 IC50 = 21 nM T87109 CM14JZ 71452176 IC50 = 114 nM T87109 CX1KZ0 71453985 IC50 = 112 nM T87109 CFGP02 71455731 IC50 = 168 nM T87109 CKT60L 71455860 Ki > 7800 nM T87109 CS27GC 71457514 IC50 = 22 nM T87109 C16OVY 71457515 IC50 = 4860 nM T87109 C3KIM9 71461149 IC50 = 22 nM T87109 CW6MK4 71462888 IC50 = 58 nM T87109 C9V6KY 71462889 IC50 = 36 nM T87109 CA3O6K 71552696 IC50 > 30000 nM T87109 C1NPL0 71552941 IC50 > 30000 nM T87109 CA4PS8 71552942 IC50 > 30000 nM T87109 C3UA9C 71553011 IC50 = 30000 nM T87109 CEZ15Y 71553012 IC50 = 2390 nM T87109 C1TR3O 71553152 IC50 = 4500 nM T87109 CHGS40 71710904 IC50 = 63.8 nM T87109 C7V5NW 73265159 IC50 = 9 nM T87109 CIJ3M8 73293373 IC50 = 237 nM T87109 C8OY6Q 76310785 IC50 = 3100 nM T87109 CAL3U7 76310788 IC50 = 1600 nM T87109 C12YAE 76314414 IC50 = 240 nM T87109 C97RBS 76317979 IC50 = 437 nM T87109 C1AI0J 76325315 IC50 = 202 nM T87109 CPQA45 76325323 IC50 = 225 nM T87109 CB5Y0Z 76332540 IC50 = 89 nM T87109 C1N6AO 76853170 IC50 = 15 nM T87109 CYE68Z 77106256 IC50 = 65 nM T87109 C0F8KW 77106257 IC50 = 33 nM T87109 C96FDY 77106258 IC50 = 23 nM T87109 CTG4Z8 77106466 IC50 = 42 nM T87109 CPO71E 77106467 IC50 = 68 nM T87109 CF9D6T 77106468 IC50 = 10 nM T87109 CJD3M8 77106469 IC50 = 56 nM T87109 CL1W2E 77106470 IC50 = 47 nM T87109 CGH13D 77106661 IC50 = 87 nM T87109 C9P7WF 77106663 IC50 = 850 nM T87109 CCSY07 77106871 IC50 = 530 nM T87109 C09OAH 77106872 IC50 = 540 nM T87109 C7EQM2 77107062 IC50 = 590 nM T87109 CGIE81 77107063 IC50 = 190 nM T87109 CJ35EI 78333498 IC50 = 335 nM T87109 C1WXC7 90644401 IC50 > 100000 nM T87109 CJ53FY 90644403 IC50 > 100000 nM T87109 CGUA74 90644405 IC50 > 100000 nM T87109 CW9Z3N 90644407 IC50 > 100000 nM T87109 CT27SY 90644409 IC50 > 100000 nM T87109 CMB4Q1 90644410 IC50 > 100000 nM T87109 CF0ZS7 90644412 IC50 > 100000 nM T87109 C1CM0J 90644414 IC50 > 100000 nM T87109 CS1Y2A 90644416 IC50 > 100000 nM T87109 CKJ16V 90644418 IC50 > 100000 nM T87109 CKH45I 90644420 IC50 > 100000 nM T87109 C3XTN6 90644422 IC50 > 100000 nM T87109 CEHV08 90644424 IC50 > 100000 nM T87109 CCR32H 90644426 IC50 > 100000 nM T87109 CA32ED 90644428 IC50 > 100000 nM T87109 CDS9Y8 90644430 IC50 > 100000 nM T87109 CEPL28 90644432 IC50 > 100000 nM T87109 C56RMJ 90644434 IC50 > 100000 nM T87109 CFW89O 90644436 IC50 > 100000 nM T87109 CY3NH1 90644438 IC50 > 100000 nM T87109 CC9FY8 90644440 IC50 > 100000 nM T87109 CYV14P 90644442 IC50 > 100000 nM T87109 CZ72JE 90655325 IC50 = 7450 nM T87109 C7VXE2 90655326 IC50 = 9310 nM T87109 CVX42T 90655327 IC50 = 4370 nM T87109 C51UDW 90655328 IC50 = 3790 nM T87109 CY8IM1 90655329 IC50 = 10110 nM T87109 CK3CL8 90655330 IC50 = 1930 nM T87109 C7GL0F 90655331 IC50 = 7380 nM T87109 C14XNE 90655332 IC50 = 1120 nM T87109 CG9O8U 90655333 IC50 = 4110 nM T87109 C82OVJ 90655334 IC50 = 5500 nM T87109 CO75LW 90655335 IC50 = 430 nM T87109 C3DC9V 90655336 IC50 = 460 nM T87109 C0Y8ZK 91933875 IC50 > 1000 nM T87109 CAU45T 91971978 IC50 > 30000 nM T87109 C2C0AG 118707521 IC50 = 439 nM T87109 C2DJA0 118707522 IC50 > 100000 nM T87109 CBF28W 118707523 IC50 > 100000 nM T87109 CQ6ON4 118707525 IC50 = 21400 nM T87109 C38UWP 118707526 IC50 > 100000 nM T87109 C64ZQX 118707543 IC50 = 66300 nM T87109 CU60YC 135431661 IC50 = 6340 nM T87109 CW0P1Q 135433657 IC50 = 1352 nM T87109 C5XIE8 136026041 IC50 = 39000 nM T87109 C5JIR2 136987005 IC50 = 5960 nM T87109 C4MJ8D 138105941 IC50 = 45 nM T87109 C3W4RO 138403252 IC50 = 3600 nM T87109 C0BSA1 145963824 IC50 = 700 nM T87109 CW05TY 145963985 IC50 = 625 nM T87109 CBT15C 145964197 IC50 = 520 nM T87109 CD9FX7 145964328 IC50 = 915 nM T87109 CPTW53 145964369 IC50 = 55 nM T87109 CN59FX 145964414 IC50 = 535 nM T87109 C3J6YH 145965218 IC50 = 215 nM T87109 CW12OV 145965254 IC50 = 50 nM T87109 CI39VD 145965319 IC50 = 175 nM T87109 C6ZW7D 145965387 IC50 = 525 nM T87109 C45SDT 145965497 IC50 = 295 nM T87109 CWK36T 145965775 IC50 = 830 nM T87109 CB8VS5 145965873 IC50 = 1155 nM T87109 C0LM9U 145966033 IC50 = 320 nM T87109 C76NKD 145966367 IC50 = 69 nM T87109 CB8J9L 145966621 IC50 = 620 nM T87109 C5D7LE 145966696 IC50 = 100 nM T87109 CMJ31A 145966880 IC50 = 1195 nM T87109 C4K2MZ 145967302 IC50 = 80 nM T87109 C6IZ1C 145967749 IC50 = 440 nM T87109 CDNC31 145967951 IC50 > 500 nM T87109 C0ZML5 145967991 IC50 = 1565 nM T87109 C5I8UB 145968214 IC50 = 175 nM T87109 CO06FU 145968732 IC50 = 1030 nM T87109 C89WUQ 145969180 IC50 = 145 nM T87109 C93CMJ 145970268 IC50 = 47 nM T87109 CD6J3O 145970533 IC50 = 50 nM T87109 CZI5A9 145970735 IC50 = 335 nM T87109 C2O1ZW 145970740 IC50 = 260 nM T87109 COG2B8 145971011 IC50 = 175 nM T87109 CK03FQ 145972343 IC50 = 200 nM T87109 CAJ0D4 145972722 IC50 = 260 nM T87109 CWB10V 145973036 IC50 = 180 nM T87109 C3P1OT 145973084 IC50 = 110 nM T87109 CG48AP 145973222 IC50 = 10 nM T87109 CYC0U9 145973723 IC50 = 825 nM T87109 CV2R6L 145973925 IC50 > 9900 nM T87109 C3UK4Q 145973964 IC50 = 610 nM T87109 CW0Y2I 145974384 IC50 = 76 nM T87109 C2YQN3 145974395 IC50 = 295 nM T87109 CH9LZ0 145974411 IC50 = 42 nM T87109 CKES90 145974470 IC50 = 4520 nM T87109 CQR37C 145974951 IC50 = 150 nM T87109 C1N0DI 145975378 IC50 = 430 nM T87109 C1PSC3 145975405 IC50 > 10000 nM T87109 CPGZ90 145975408 IC50 = 54 nM T87109 CWF6C7 145976053 IC50 = 185 nM T87109 CSH68V 145976072 IC50 = 230 nM T87109 C43TWQ 145976109 IC50 = 520 nM T87109 C18QUZ 145976185 IC50 = 4010 nM T87109 CY2IN5 145976421 IC50 = 53 nM T87109 C9T0SR 145976580 EC50 = 1470 nM T87109 CUP7F4 145976617 IC50 = 160 nM T87109 CLI3T5 145977030 IC50 = 245 nM T87109 CGV9W7 145977170 IC50 = 230 nM T87109 CJ2UR4 145977480 IC50 = 1120 nM T87109 CA7S8J 145977657 IC50 > 10000 nM T87109 CU5L2G 145977991 IC50 > 10000 nM T87109 CMG04P 145978001 IC50 = 48 nM T87109 CS3ID1 145978144 IC50 = 1180 nM T87109 C2MD1Q 155513187 IC50 > 10000 nM T87109 CY18OB 155538177 IC50 = 354 nM T87109 CD2LG1 155541831 IC50 = 1030 nM T87109 D00ERW 44444843 Ki > 7826 nM T87109 D00HVA 11624601 Ki > 7800 nM T87109 D00JGL 6419753 IC50 = 171 nM T87109 D06QYR 53472153 IC50 = 32 nM T87109 D0A7FQ 11644425 IC50 = 510 nM T87109 D0F0AX 135413546 IC50 = 35 nM T87109 D0H4VB 71461150 IC50 = 59 nM T87109 D0L4WN 31420 IC50 = 330 nM T87109 D0ME9B 46868971 IC50 > 10 nM T87109 D0N3LC 90643548 IC50 = 104 nM T87109 D0O6OH 71553154 IC50 = 110 nM T87109 D0Q3NG 11715520 Ki > 7800 nM T87109 D0RJ8J 76072859 IC50 = 84 nM T87109 D0S7IE 11658882 Ki > 7800 nM T87109 D0UN8H 5288600 IC50 = 1000 nM T87109 D0VC0I 5169 IC50 = 188 nM T87109 D0Y6OK 6688 IC50 > 40000 nM T64795 D0F4GF 24765479 IC50 = 1.2 nM T64795 D0W8XT 60663 IC50 = 200 nM T64795 CMT3P0 480764 IC50 = 1000 nM T64795 C79YAJ 1034176 IC50 = 1560 nM T64795 CUQ4R7 2987239 IC50 > 10000 nM T64795 C1TY4I 3239035 IC50 = 3110 nM T64795 C39ETP 3243445 IC50 = 11390 nM T64795 C0F8EP 3519901 IC50 = 1000 nM T64795 C72QNV 3596240 IC50 = 2080 nM T64795 CY4OJ0 3596497 IC50 = 11370 nM T64795 CY1C6K 4124732 IC50 = 1160 nM T64795 C6US3T 4124734 IC50 = 1410 nM T64795 C6UI5J 4124736 IC50 = 4690 nM T64795 CU57CD 4597377 IC50 = 53500 nM T64795 CNZ1F7 6458316 IC50 = 1140 nM T64795 CP5NF6 6461757 IC50 = 170 nM T64795 CO4F3A 6616145 IC50 = 2530 nM T64795 CQM3D8 6616154 IC50 = 1100 nM T64795 C8AXC9 7189282 IC50 = 11380 nM T64795 CEH68S 7189284 IC50 = 12330 nM T64795 CR4KG1 10323629 IC50 = 1020 nM T64795 CGSI34 10411835 IC50 = 1530 nM T64795 CK08WH 11167614 IC50 = 2500 nM T64795 CUPN76 11201837 IC50 = 35800 nM T64795 C6P4JC 11348836 IC50 = 10700 nM T64795 CJ2E6Z 11476189 IC50 = 21577.44 nM T64795 CN0OL7 15262444 IC50 = 27669.42 nM T64795 CG8KR9 16005860 IC50 = 43 nM T64795 CXL7Z2 16046181 IC50 = 450 nM T64795 CL17AW 16126700 IC50 = 100 nM T64795 COK8Y4 16215108 IC50 = 930 nM T64795 C3PO4X 16216102 IC50 = 1010 nM T64795 C83HGX 23653556 IC50 = 3310 nM T64795 C85MEH 24782219 IC50 = 1840 nM T64795 C2P6ZS 24782229 IC50 = 5820 nM T64795 C4PVE2 24782723 IC50 = 14120 nM T64795 CJS73W 24784770 IC50 = 22780 nM T64795 C7NVW3 24785007 IC50 = 14860 nM T64795 CMUP43 24785249 IC50 = 8520 nM T64795 C7Z9DM 24785508 IC50 = 5820 nM T64795 CQ30ZC 24785510 IC50 = 1520 nM T64795 C6P9NV 24785782 IC50 = 960 nM T64795 CYM79T 24786041 IC50 = 2070 nM T64795 CN8E4M 24786051 IC50 = 1930 nM T64795 C7P4SR 24804568 IC50 = 7980 nM T64795 CAV92J 25112129 IC50 = 2269.86 nM T64795 CL03EY 25112130 IC50 = 369.83 nM T64795 CM61YC 25112244 IC50 = 339.63 nM T64795 CSP58A 25112245 IC50 = 1199.5 nM T64795 C6K9PN 25112246 IC50 = 4539.42 nM T64795 CG9M6A 25112247 IC50 = 139.96 nM T64795 CO6BI7 25112354 IC50 = 9162.2 nM T64795 CN9Q1A 25112356 IC50 = 5840 nM T64795 CF36CS 25112467 IC50 = 230 nM T64795 CJE9H5 25112468 IC50 = 169.82 nM T64795 C7C4GE 25168962 IC50 = 2610 nM T64795 CLOS63 25168963 IC50 = 2780 nM T64795 CSZ0A2 25168964 IC50 = 1800 nM T64795 CUJ69G 25168965 IC50 = 3270 nM T64795 CQ82ZP 25168966 IC50 = 4210 nM T64795 CPV5L9 25168967 IC50 = 3340 nM T64795 CW1MH2 25169093 IC50 = 3810 nM T64795 CAQ9X2 25169094 IC50 = 3140 nM T64795 CN6PE2 25169095 IC50 = 1480 nM T64795 CE2Z7S 25169096 IC50 = 280 nM T64795 CJ40DP 25169097 IC50 = 750 nM T64795 C15BYF 25169098 IC50 = 2400 nM T64795 CT7AO0 25169361 IC50 = 1910 nM T64795 C45NJD 25169363 IC50 = 2440 nM T64795 CEL93W 25169364 IC50 = 1810 nM T64795 C8VCL4 25169493 IC50 = 3400 nM T64795 CMC75E 25169494 IC50 = 2910 nM T64795 C6NA1J 25194889 IC50 = 8.17 nM T64795 C5XDE0 25195536 IC50 = 190 nM T64795 C3GX5Y 25221039 IC50 = 3710 nM T64795 C64MWD 25221145 IC50 = 420 nM T64795 CS87VL 25221147 IC50 = 2320 nM T64795 C6WJ5R 25221148 IC50 = 360 nM T64795 CN57OJ 25221261 IC50 = 1540 nM T64795 C2ON7I 25221262 IC50 = 1670 nM T64795 CW8ZD6 25221263 IC50 = 16100 nM T64795 CR8DL9 25221264 IC50 = 600 nM T64795 CM4P7I 25221265 IC50 = 280 nM T64795 CA26GP 25221368 IC50 = 1020 nM T64795 C60RHJ 30634189 IC50 = 1080 nM T64795 C1REU6 35537998 IC50 = 41 nM T64795 CPS3Z2 44392185 IC50 = 299.92 nM T64795 CUM41S 44416823 IC50 = 24154.61 nM T64795 CB5T1D 44417094 IC50 = 1130 nM T64795 CVC70A 44417099 IC50 = 2040 nM T64795 C8QAM5 44417106 IC50 = 1480 nM T64795 CM8P0A 44417111 IC50 = 1610 nM T64795 C0TJ4W 44417112 IC50 = 1330 nM T64795 CO2N5A 44417143 IC50 = 2130 nM T64795 C4HO2I 44417148 IC50 = 1390 nM T64795 C8JQ0A 44417174 IC50 = 990 nM T64795 C3CTO5 44417176 IC50 = 1220 nM T64795 C41VLE 44417195 IC50 = 1860 nM T64795 CY58AR 44417212 IC50 = 2180 nM T64795 C4ODB3 44417219 IC50 = 2750 nM T64795 C4RM3Y 44422184 IC50 = 5970 nM T64795 CCZ87N 44422276 IC50 = 2790 nM T64795 C8W2UY 44422328 IC50 = 7960 nM T64795 C8VX5M 44422330 IC50 = 4630 nM T64795 C6NV3B 44422568 IC50 = 2040 nM T64795 CQEX93 44422611 IC50 = 2020 nM T64795 C6FW4I 44423577 IC50 = 1010 nM T64795 C1UJ8C 44423580 IC50 = 4470 nM T64795 C16ZOD 44423582 IC50 = 3630 nM T64795 C5P6NC 44423583 IC50 = 3490 nM T64795 CPYR60 44423585 IC50 = 6010 nM T64795 C79QBV 44423587 IC50 = 2640 nM T64795 C84SAP 44423593 IC50 = 3520 nM T64795 C4UBT2 44423595 IC50 = 370 nM T64795 CG7M1W 44423598 IC50 = 2730 nM T64795 C1I5ZF 44423607 IC50 = 1670 nM T64795 CZVY86 44438773 IC50 = 2030 nM T64795 C92ZRU 44438777 IC50 = 1810 nM T64795 C65SUA 44438796 IC50 = 3530 nM T64795 C5UHB1 44438807 IC50 = 8880 nM T64795 CG6JK1 44438810 IC50 = 4090 nM T64795 C2XAI7 44438814 IC50 = 8280 nM T64795 C7ZXI2 44438821 IC50 = 5250 nM T64795 C6VBZ3 44438823 IC50 = 1620 nM T64795 CI80QX 44577778 IC50 = 250 nM T64795 CX7HN8 44577815 IC50 = 100 nM T64795 C6G3JA 44577816 IC50 = 190 nM T64795 C5CTS6 44577817 IC50 = 880 nM T64795 CAF21G 44577856 IC50 = 250 nM T64795 CQ20ZL 44577857 IC50 = 53.02 nM T64795 CG8CD3 44577858 IC50 = 340 nM T64795 C3U8JW 44577859 IC50 = 260 nM T64795 CXJ8A9 44577924 IC50 = 740 nM T64795 CX60LY 44577925 IC50 = 980 nM T64795 CYT60I 44577926 IC50 = 1110 nM T64795 CKV0C9 44577927 IC50 = 280 nM T64795 C5LJ0D 44577963 IC50 = 95 nM T64795 CT4A5Y 44577964 IC50 = 480 nM T64795 CV75CM 44577965 IC50 = 320 nM T64795 CNR6Q0 44577966 IC50 = 390 nM T64795 CW59ZQ 46224946 IC50 = 429.54 nM T64795 CD56HO 46224947 IC50 = 868.96 nM T64795 CF29RU 46224974 IC50 = 2167.7 nM T64795 C4FNT2 46225003 IC50 = 1009.25 nM T64795 C3XS1U 46225137 IC50 = 12705.74 nM T64795 C19ZCY 46861765 IC50 = 1230 nM T64795 CTE2S8 46861766 IC50 = 2080 nM T64795 C6AH4P 46887649 IC50 = 4000 nM T64795 CO2PM3 46887855 IC50 = 3170 nM T64795 C28HMC 46888212 IC50 = 2390 nM T64795 CY3PF5 46888270 IC50 = 1470 nM T64795 CUI8G5 46888332 IC50 = 12600 nM T64795 CK2R1Z 46911114 IC50 = 650 nM T64795 CIE3S8 48830232 IC50 = 2200 nM T64795 CXV8O9 49798178 IC50 = 9200 nM T64795 CJPX96 49798179 IC50 = 2100 nM T64795 CGVY07 49798180 IC50 = 1940 nM T64795 CGZU79 49798181 IC50 = 1300 nM T64795 C64RGL 49798202 IC50 = 1710 nM T64795 CI2S3D 49798203 IC50 = 2220 nM T64795 CW2MV4 49798204 IC50 = 2220 nM T64795 C07YMH 49798225 IC50 = 16130 nM T64795 C6WML9 49798226 IC50 = 3030 nM T64795 C65UBA 49798227 IC50 = 3210 nM T64795 C87MZA 49798250 IC50 = 2800 nM T64795 C5R7BC 49798251 IC50 = 1750 nM T64795 C6H3ZK 49798252 IC50 = 1310 nM T64795 CHF38W 49798253 IC50 = 8750 nM T64795 CK68OE 49798275 IC50 = 1190 nM T64795 CY2SA7 49798276 IC50 = 130010 nM T64795 CS57TO 49798310 IC50 = 7250 nM T64795 C8QJ2T 49798338 IC50 = 1780 nM T64795 C1Z3VU 49798339 IC50 = 3020 nM T64795 C5TSJ7 49798341 IC50 = 7470 nM T64795 C7Y5HN 49798582 IC50 = 10250 nM T64795 C0O3RW 49798584 IC50 = 3350 nM T64795 C47XQP 49798585 IC50 = 7080 nM T64795 CJ3T5A 49798606 IC50 = 4370 nM T64795 C4XUW2 49798607 IC50 = 1450 nM T64795 C3YXT8 49798608 IC50 = 2820 nM T64795 CQM71L 49798609 IC50 = 4300 nM T64795 CUDE92 50898773 IC50 = 41 nM T64795 C2HJL6 50942025 IC50 = 860 nM T64795 CA75HL 51050194 IC50 = 8800 nM T64795 C9P4YV 53316457 IC50 = 1730 nM T64795 CW7TF1 53316459 IC50 = 2480 nM T64795 CPS12B 53317097 IC50 = 89 nM T64795 CUR97Z 53324407 IC50 = 21150 nM T64795 C4ZO1H 53324408 IC50 = 1290 nM T64795 C7OJ6G 53325710 IC50 = 17050 nM T64795 CH5A9S 53484202 IC50 = 7310 nM T64795 C8C5PV 54752457 IC50 = 36 nM T64795 CE4L6S 54752459 IC50 = 85 nM T64795 CDON72 56658273 IC50 = 1200 nM T64795 CC6J9O 56658274 IC50 = 320 nM T64795 CG1XF2 56658275 IC50 = 370 nM T64795 CL36UH 56658276 IC50 = 89 nM T64795 C6GIK1 56658277 IC50 = 260 nM T64795 C7RGZ8 56658278 IC50 = 130 nM T64795 C3MFK4 56658279 IC50 = 180 nM T64795 CIP1C9 56658280 IC50 = 770 nM T64795 C67LRT 56661771 IC50 = 240 nM T64795 CW9K5P 56661772 IC50 = 130 nM T64795 CJ4V1H 56661773 IC50 = 90 nM T64795 CAPH84 56661774 IC50 = 140 nM T64795 CGB20Q 56665221 IC50 = 82 nM T64795 CQ6M2B 56665222 IC50 = 170 nM T64795 C0QOY7 56666255 IC50 = 4180 nM T64795 CYQM41 56668677 IC50 = 510 nM T64795 CUIF48 56668678 IC50 = 860 nM T64795 CN90RO 56672151 IC50 = 3000 nM T64795 CX25FY 56672152 IC50 = 2000 nM T64795 CM92CD 56672153 IC50 = 750 nM T64795 CU8OE1 56672154 IC50 = 120 nM T64795 CDP35F 56672155 IC50 = 200 nM T64795 CI3T9O 56675544 IC50 = 130 nM T64795 C6Q2IP 56678875 IC50 = 220 nM T64795 CML96V 56678876 IC50 = 1200 nM T64795 CHB86Q 56678877 IC50 = 94 nM T64795 C0FI2Q 56682190 IC50 = 390 nM T64795 CPTW59 56682191 IC50 = 250 nM T64795 CHU51L 66549542 IC50 = 15500 nM T64795 CVUT64 66549717 IC50 = 480 nM T64795 CAV5N8 66549719 IC50 = 4230 nM T64795 C1MDS9 66549721 IC50 = 760 nM T64795 C5TNE0 66551172 IC50 = 2580 nM T64795 CBI4P9 66551368 IC50 = 230 nM T64795 CHL24B 66551569 IC50 = 12000 nM T64795 CCH8K4 66551570 IC50 = 2100 nM T64795 C3SCF6 66551759 IC50 = 100 nM T64795 CY74BK 71570778 IC50 = 1790 nM T64795 C6WFT5 71570924 IC50 = 1270 nM T64795 C8C9ZP 71660493 IC50 = 320 nM T64795 C02RPG 71660495 IC50 = 310 nM T64795 CW7TD2 71716405 IC50 = 1420 nM T64795 CL7GF4 72724691 IC50 = 310 nM T64795 C8NQH6 72724692 IC50 = 550 nM T64795 CJAF45 72724694 IC50 = 460 nM T64795 CCOZ75 72725613 IC50 = 390 nM T64795 CLXH36 72793718 IC50 = 2100 nM T64795 CDM04P 76310604 IC50 = 3260 nM T64795 CA83KU 76314239 IC50 = 1360 nM T64795 C3TXQ5 76321521 IC50 = 654 nM T64795 CP9V7B 76328692 IC50 = 3240 nM T64795 C2YIP6 76332364 IC50 = 56 nM T64795 CNA06U 76332366 IC50 = 2650 nM T64795 CF7GZ5 86292750 IC50 = 2730 nM T64795 CF7Y2I 86292753 IC50 = 11030 nM T64795 CV8OI5 86292754 IC50 = 4760 nM T64795 CDV37Y 86292938 IC50 = 5910 nM T64795 CEPV50 90655094 IC50 = 1810 nM T64795 CUD8W4 90655095 IC50 = 730 nM T64795 CV21UB 90655097 IC50 = 600 nM T64795 CCL46V 90655099 IC50 = 1040 nM T64795 C0JTE3 90655100 IC50 = 520 nM T64795 CEJK10 92135927 IC50 = 5650 nM T64795 CG60JW 117700665 IC50 = 10080 nM T64795 C48PFK 118512802 IC50 = 3200 nM T64795 CLHP58 118560158 IC50 = 4.2 nM T64795 C9S4YL 118560191 IC50 = 3.1 nM T64795 C0LR9M 118560290 IC50 = 3.2 nM T64795 C7Y8FJ 118560322 IC50 = 7 nM T64795 CE6O4V 118560356 IC50 = 11 nM T64795 CMAN70 118560393 IC50 = 12 nM T64795 C4VG3F 118560394 IC50 = 6.8 nM T64795 CZ6O0E 118560399 IC50 = 2.2 nM T64795 CVRO18 118560401 IC50 = 1.1 nM T64795 CZ62GY 118560409 IC50 = 1.5 nM T64795 CL12OZ 118560423 IC50 = 2.5 nM T64795 CH84UX 118560458 IC50 = 4.3 nM T64795 C7Y2LQ 118560466 IC50 = 15 nM T64795 C0JAX6 118560472 IC50 = 23 nM T64795 CDJL48 118560488 IC50 = 1.9 nM T64795 CY2KI3 118560543 IC50 = 4.6 nM T64795 C37PDX 118560579 IC50 = 7.1 nM T64795 CG25JS 118560588 IC50 = 2.3 nM T64795 CLK32A 118560592 IC50 = 1.4 nM T64795 C04FRX 118560613 IC50 = 1.4 nM T64795 CB41MH 118560618 IC50 = 6.4 nM T64795 CS0RQ3 118560699 IC50 = 2.8 nM T64795 CQG3K7 118560709 IC50 = 1 nM T64795 C2DA9Z 118962193 IC50 = 3.5 nM T64795 CB56CV 122189312 IC50 = 7400 nM T64795 CL15MQ 122189314 IC50 = 2500 nM T64795 C1PRY5 122189316 IC50 = 1900 nM T64795 C4EF6B 122189318 IC50 = 2400 nM T64795 CX35ZS 122189320 IC50 = 6400 nM T64795 CZ16JP 122189321 IC50 = 5200 nM T64795 CF6D2P 126740597 IC50 = 1.1 nM T64795 CAYS28 126740598 IC50 = 10 nM T64795 CIQ23U 126740608 IC50 = 1.1 nM T64795 C1O5VB 126740610 IC50 = 2.3 nM T64795 C9KEY6 126740618 IC50 = 2.6 nM T64795 CA1M2Q 126740623 IC50 = 3.4 nM T64795 CNUF36 126740624 IC50 = 1.3 nM T64795 COE64S 126740626 IC50 = 2.2 nM T64795 CS2Y3W 126740650 IC50 = 3.4 nM T64795 CHO17P 126740652 IC50 = 2.4 nM T64795 CKNV98 126740697 IC50 = 3.5 nM T64795 C0AI1V 132991411 IC50 = 142 nM T64795 C1XR9I 134130259 IC50 = 193 nM T64795 C3P7TZ 134130807 IC50 = 42 nM T64795 C9RZB3 134131854 IC50 = 178 nM T64795 CW0Q7I 134132801 IC50 = 76 nM T64795 CHR09A 134133339 IC50 = 107 nM T64795 CG21YN 134133529 IC50 = 304 nM T64795 CE32KO 134133599 IC50 = 18 nM T64795 CH9MI7 134133901 IC50 = 370 nM T64795 C3GIH1 134134030 IC50 = 25 nM T64795 CEWV89 134134318 IC50 = 8 nM T64795 C5RY7Q 134134580 IC50 = 26 nM T64795 CBC5I3 134135133 IC50 = 211 nM T64795 C67QGZ 134135164 IC50 = 5 nM T64795 CV0I4O 134135871 IC50 = 7 nM T64795 CJM8S0 134135899 IC50 = 40 nM T64795 CQ54CZ 134135912 IC50 = 227 nM T64795 CK9MG1 134136380 IC50 = 29 nM T64795 CJ4T0C 134138248 IC50 = 6070 nM T64795 CW4BU5 134138250 IC50 = 115 nM T64795 CLW07U 134138308 IC50 = 140 nM T64795 CERI05 134138759 IC50 = 4 nM T64795 C29IBJ 134139406 IC50 = 441 nM T64795 CPG8R2 134139460 IC50 > 7260 nM T64795 CRJ72V 134140275 IC50 = 27 nM T64795 C9CO2P 134140278 IC50 = 45 nM T64795 C39PGW 134140468 IC50 = 576 nM T64795 CWI1J7 134140478 IC50 = 12360 nM T64795 C8L5VZ 134140864 IC50 = 4 nM T64795 C62AVQ 134141003 IC50 = 40 nM T64795 C3NRL2 134141387 IC50 = 37 nM T64795 CIPG12 134141754 IC50 > 8500 nM T64795 C90WMC 134141766 IC50 = 390 nM T64795 CR29YW 134141773 IC50 = 65 nM T64795 C4IV9M 134141806 IC50 > 5300 nM T64795 CGA34U 134141893 IC50 = 613 nM T64795 C6U2PJ 134142122 IC50 = 47 nM T64795 C0CT2A 134142164 IC50 = 23 nM T64795 CVC5M6 134142399 IC50 = 360 nM T64795 CXK8D7 134142518 IC50 = 13 nM T64795 C16TWR 134142614 IC50 = 188 nM T64795 C2VSP7 134143155 IC50 = 29 nM T64795 CQ80GN 134143440 IC50 = 68 nM T64795 C1PT9H 134143519 IC50 = 17 nM T64795 CEG7S4 134143554 IC50 = 16 nM T64795 CH03BE 134143575 IC50 = 57 nM T64795 C2VJ7N 134143801 IC50 > 9400 nM T64795 C9A1XL 134143901 IC50 = 6280 nM T64795 CS7G2P 134144179 IC50 = 79 nM T64795 C1OLQ9 134144496 IC50 = 262 nM T64795 C8XR0U 134145066 IC50 = 196 nM T64795 CN8WV9 134145759 IC50 = 15 nM T64795 C6OD8Y 134145781 IC50 = 12 nM T64795 CB6QF0 134145994 IC50 = 31 nM T64795 C7GL6O 134146020 IC50 = 38 nM T64795 CY5ME7 134146171 IC50 = 45 nM T64795 CG7RX1 134146440 IC50 = 582 nM T64795 CN2ST6 134146817 IC50 > 10000 nM T64795 CE15VD 134146997 IC50 = 25 nM T64795 CV73DS 134147142 IC50 = 457 nM T64795 CU0WK1 134147287 IC50 = 875 nM T64795 C1JXF2 134147318 IC50 = 34 nM T64795 C6J0RP 134147643 IC50 = 627 nM T64795 CHN1C9 134147829 IC50 = 12710 nM T64795 C0ZQM8 134147890 IC50 = 476 nM T64795 C5C7BZ 134147980 IC50 = 754 nM T64795 C9W1AN 134148285 IC50 = 293 nM T64795 CW9M8G 134148369 IC50 = 35 nM T64795 C45XMS 134148468 IC50 = 8 nM T64795 C20MDR 134148760 IC50 = 78 nM T64795 CWZ47K 134149196 IC50 = 13 nM T64795 C1UY6K 134149672 IC50 = 6 nM T64795 CYQ43A 134149751 IC50 = 420 nM T64795 C4FC6U 134149941 IC50 = 13 nM T64795 CJZ29K 134149992 IC50 > 10000 nM T64795 CML57E 134151608 IC50 = 53 nM T64795 CO1JA4 134151710 IC50 = 279 nM T64795 CV25WH 134151973 IC50 = 605 nM T64795 C0NU4T 134152220 IC50 = 24 nM T64795 CVLO27 134152587 IC50 = 26 nM T64795 C7TV2H 134152703 IC50 = 597 nM T64795 CKI47N 134152745 IC50 = 305 nM T64795 C7NV2W 134152994 IC50 = 108 nM T64795 CFK81J 134153093 IC50 = 676 nM T64795 C19LMT 134153241 IC50 = 33 nM T64795 CZX13T 134153284 IC50 = 256 nM T64795 CV9ME7 134153508 IC50 = 7 nM T64795 C4L8QS 134153676 IC50 = 6110 nM T64795 C0V6YF 134153738 IC50 = 47 nM T64795 CEA6H8 134153757 IC50 = 286 nM T64795 CMH28S 134154353 IC50 = 187 nM T64795 C3AW2M 134155076 IC50 = 1139 nM T64795 CX8P0D 134155552 IC50 = 102 nM T64795 CN98ZC 134156036 IC50 > 10000 nM T64795 CAS9U3 134156465 IC50 = 220 nM T64795 CE8V5G 134156616 IC50 = 260 nM T64795 C9F3EG 134156994 IC50 = 36 nM T64795 CS4PX9 134157075 IC50 > 10000 nM T64795 C5TC7R 134157194 IC50 = 20 nM T64795 CLMT10 134157774 IC50 = 23 nM T64795 C5XSK9 135462545 IC50 = 560 nM T64795 CSA5U4 135906464 IC50 = 679.2 nM T64795 C13SAP 135906465 IC50 = 159.96 nM T64795 CSJ58R 135960710 IC50 = 570 nM T64795 CY60FR 135971402 IC50 = 1840.77 nM T64795 CIS69U 135971403 IC50 = 2018.37 nM T64795 CV9XI2 135971413 IC50 = 3126.08 nM T64795 C05KZL 141634203 IC50 = 45 nM T64795 CN9O6Q 145963763 IC50 = 87 nM T64795 CBC6A4 145964052 IC50 = 230 nM T64795 CZFE02 145964073 IC50 = 14 nM T64795 C6WB0E 145964120 IC50 = 55 nM T64795 C1RJ5L 145964213 IC50 = 82 nM T64795 C7TAQ5 145964444 IC50 = 5700 nM T64795 CL3J5T 145964488 IC50 = 250 nM T64795 CX7TC4 145964712 IC50 = 55 nM T64795 C0JGD5 145964736 IC50 = 28 nM T64795 CUQD06 145964872 IC50 = 1000 nM T64795 C6V5PA 145965039 IC50 = 250 nM T64795 CSJV78 145965046 IC50 = 44 nM T64795 CEK7F5 145965051 IC50 = 58 nM T64795 CU79FE 145965065 IC50 = 35 nM T64795 C3XZ9G 145965167 IC50 = 11 nM T64795 CZ7VP8 145965333 IC50 = 53 nM T64795 COA0D4 145965395 IC50 = 70 nM T64795 CG5D0A 145965520 IC50 = 250 nM T64795 C2SV8D 145965539 IC50 = 59 nM T64795 CB24MN 145965576 IC50 = 180 nM T64795 C8MUI9 145965686 IC50 = 240 nM T64795 CM0C4Q 145965785 IC50 = 240 nM T64795 C74GDJ 145965861 IC50 = 52 nM T64795 CSR0W9 145965878 IC50 = 1150 nM T64795 CP9GX0 145965960 IC50 = 220 nM T64795 CC25LD 145966135 IC50 = 17 nM T64795 CY6NH0 145966175 IC50 = 380 nM T64795 C6P5GM 145966272 IC50 = 46 nM T64795 C7MOG0 145966280 IC50 = 180 nM T64795 CNG80S 145966315 IC50 = 1400 nM T64795 C3I5WD 145966882 IC50 > 10000 nM T64795 CB6G2J 145966887 IC50 = 88 nM T64795 C9OZ7B 145966987 IC50 > 10000 nM T64795 CQ6S4I 145967128 IC50 = 140 nM T64795 CIFN68 145967321 IC50 = 6.2 nM T64795 C3P6KV 145967526 IC50 = 6.5 nM T64795 CWRS54 145967754 IC50 = 335 nM T64795 C9GYA8 145968219 IC50 = 410 nM T64795 C3F9UM 145968918 IC50 = 88 nM T64795 CO1FC6 145968951 IC50 = 160 nM T64795 C8A3JX 145968953 IC50 = 5.1 nM T64795 CX2Q3S 145969169 IC50 = 170 nM T64795 C93RXD 145970771 IC50 > 10000 nM T64795 CJE56F 145971412 IC50 = 4.5 nM T64795 CXMQ72 145971782 IC50 = 190 nM T64795 CM92KQ 145971885 IC50 = 510 nM T64795 CK06VY 145972088 IC50 = 210 nM T64795 CO0FR7 145972093 IC50 = 110 nM T64795 CAOS28 145973012 IC50 = 180 nM T64795 C2C1ST 145973030 IC50 = 310 nM T64795 CQYB38 145973089 IC50 = 14 nM T64795 C8UN1L 145973107 IC50 = 460 nM T64795 C2L7RP 145973300 IC50 = 200 nM T64795 CQ7WG9 145973409 IC50 = 98 nM T64795 C1N4UG 145973443 IC50 = 330 nM T64795 CHZ21U 145973703 IC50 = 280 nM T64795 CH9P2S 145973704 IC50 = 490 nM T64795 CHQ32U 145973751 IC50 = 460 nM T64795 C5OX8I 145973789 IC50 = 34 nM T64795 CON93L 145973912 IC50 = 13 nM T64795 CM78OR 145974461 IC50 = 71 nM T64795 C7B2VG 145974480 IC50 = 920 nM T64795 C8G1KM 145974485 IC50 = 480 nM T64795 CED15B 145974511 IC50 = 250 nM T64795 C2OL7I 145975061 IC50 = 540 nM T64795 C9UVC6 145975140 IC50 = 2.2 nM T64795 CDB4P8 145975231 IC50 = 870 nM T64795 CR2N8T 145975397 IC50 = 18 nM T64795 C58WOB 145975751 IC50 = 54 nM T64795 C3W2OE 145975832 IC50 = 240 nM T64795 CMWY20 145975926 IC50 = 360 nM T64795 C1YSW7 145976102 IC50 = 260 nM T64795 CK8X4G 145976223 IC50 = 2360 nM T64795 CO8KN3 145976268 IC50 = 45 nM T64795 CN72ZM 145976351 IC50 = 3700 nM T64795 C4KF1L 145976387 IC50 = 320 nM T64795 C3XE5S 145976394 IC50 = 22 nM T64795 CE50WI 145976410 IC50 = 530 nM T64795 CGA1B5 145976660 IC50 = 350 nM T64795 C2BVH9 145976792 IC50 = 760 nM T64795 C1QU0T 145976799 IC50 = 910 nM T64795 CM6ZT8 145976855 IC50 = 45 nM T64795 CLCM81 145976857 IC50 = 120 nM T64795 C1L2NM 145977186 IC50 = 54 nM T64795 C0S3TG 145977189 IC50 = 130 nM T64795 CH3FM6 145977296 IC50 = 24 nM T64795 CAR4F9 145977337 IC50 = 200 nM T64795 C5I6VA 145977340 IC50 = 17 nM T64795 C21VED 145977676 IC50 = 600 nM T64795 CU38DI 145977733 IC50 = 32 nM T64795 CSE52C 145977745 IC50 = 320 nM T64795 C45HOF 145977787 IC50 = 3.4 nM T64795 C1XD8F 145977860 IC50 = 60 nM T64795 CCL06J 145977910 IC50 = 20 nM T64795 CI89TQ 145978258 IC50 = 100 nM T64795 C8BD3R 145978287 IC50 = 49 nM T64795 C7DV6A 145978317 IC50 = 5 nM T64795 CL36DE 145978466 IC50 = 35 nM T64795 CU0N4O 145978657 IC50 = 8.1 nM T64795 CGW6Q5 145978668 IC50 = 200 nM T64795 CV4LT9 153635960 IC50 = 5130 nM T64795 C8ET9R 155524767 EC50 = 12480 nM T64795 D02DDI 11964508 IC50 = 960 nM T64795 D02DUO 9980573 IC50 = 900 nM T64795 D02SSG 25112470 IC50 = 4200 nM T64795 D03HCT 25196629 IC50 = 16870 nM T64795 D05MYH 44568140 IC50 = 1039.92 nM T64795 D06EPZ 25196850 IC50 = 3720 nM T64795 D06FWY 44416787 IC50 = 1119.44 nM T64795 D06ORM 44567629 IC50 = 349.95 nM T64795 D06UAX 16048644 IC50 = 260 nM T64795 D07UBR 44417210 IC50 = 1010 nM T64795 D09QCD 44567628 IC50 = 380 nM T64795 D0JO8Q 44416758 IC50 = 4102.04 nM T64795 D0K5RX 135401968 IC50 = 130 nM T64795 D0K9NK 16066792 IC50 = 1520 nM T64795 D0M2EZ 10416322 IC50 = 110 nM T64795 D0N5RQ 10031616 IC50 = 250 nM T64795 D0QM9Y 25196851 IC50 = 1950 nM T64795 D0R5FO 44568141 IC50 = 630 nM T64795 D0S5QB 44342044 IC50 = 13031.67 nM T64795 D0T6NE 44540045 IC50 = 37 nM T64795 D0V3NI 44416844 IC50 = 4581.42 nM T64795 D0V9CG 44422402 IC50 = 2460 nM T64795 D0VE0Q 72936 IC50 = 1000 nM T64795 D0X3HB 25196630 IC50 = 9230 nM T64795 D0X7VM 23661603 IC50 = 41 nM T64795 D0Y4WI 44422187 IC50 = 3380 nM T64795 D0Z4JL 25196743 IC50 = 2080 nM T86702 D00HNB 25419 IC50 = 300000 nM T86702 D00MDP 466151 Ki = 0.27 nM T86702 D04AIT 5280445 IC50 = 16200 nM T86702 D05EJG 6305 IC50 > 500000 nM T86702 D0K8KX 5280343 IC50 = 5570 nM T86702 D0S0LZ 54671203 IC50 = 25000 nM T86702 D05VZE 119031 Ki = 2.4 nM T86702 D0MW3H 9824350 Ki = 56 nM T86702 D0N4IV 10718956 IC50 > 1000 nM T86702 D0G1LL 74221072 IC50 > 100000 nM T86702 D0N6ZA 74221131 IC50 > 100000 nM T86702 D0UM5R 74221070 IC50 = 13000 nM T86702 D00UCC 9827497 IC50 = 12 nM T86702 D01DVX 9847838 IC50 = 285 nM T86702 D03BOZ 3342298 IC50 = 7.1 nM T86702 D05VNG 9908389 IC50 = 12 nM T86702 D08CEE 10478364 Ki = 310 nM T86702 D0E5GY 9904965 Ki = 310 nM T86702 D0P8YC 5362422 IC50 = 0.56 nM T86702 D0Q1CD 6918336 IC50 = 134 nM T86702 D0T2IQ 443600 IC50 = 6000 nM T86702 D0T9HG 132519 IC50 = 1.9 nM T86702 D0Y1XT 128564 Ki < 10 nM T86702 CNA81R 1836 IC50 = 2000 nM T86702 CY78XM 4218 Ki = 18 nM T86702 CFY8Q2 4230 IC50 = 18 nM T86702 CE85VA 68310 IC50 > 500000 nM T86702 CZ06IH 70878 Ki = 33000 nM T86702 C04KYL 83169 Ki = 8000 nM T86702 CES96Q 98767 Ki = 84000 nM T86702 CKUP25 101176 Ki = 2100 nM T86702 COZ0S7 111050 IC50 = 500000 nM T86702 C1HS6D 117439 IC50 = 500000 nM T86702 CXO86G 154135 IC50 = 1060 nM T86702 CDJS43 154136 IC50 = 33 nM T86702 C50IPY 154137 IC50 = 41 nM T86702 C7ROG5 177347 IC50 = 7950 nM T86702 CJ62BZ 193987 IC50 = 527 nM T86702 C9RXD1 439917 IC50 = 500000 nM T86702 C0ITQ9 444789 Ki = 19 nM T86702 CV60YH 445010 IC50 = 19 nM T86702 CK9M3P 445018 IC50 = 3.1 nM T86702 CQ7G0V 446065 Ki = 2 nM T86702 CBTK84 446505 IC50 = 30000 nM T86702 C4D7TS 448002 Ki = 131.83 nM T86702 CR51PG 448593 Ki = 229.09 nM T86702 C9I8WB 478379 Ki = 9 nM T86702 C39BCA 675678 IC50 > 500000 nM T86702 CW39GN 700653 IC50 = 500000 nM T86702 CHIO49 700663 Ki = 71000 nM T86702 CP1Q6R 703233 IC50 = 77000 nM T86702 CGSY63 706490 IC50 = 500000 nM T86702 CRF9Z4 707055 IC50 = 190000 nM T86702 C7Z0ES 712438 Ki = 18000 nM T86702 CZM23W 736160 Ki = 356000 nM T86702 CF2N6B 830422 IC50 = 97000 nM T86702 C3ML4O 853750 IC50 > 500000 nM T86702 C26JCX 853880 IC50 = 500000 nM T86702 CE6FN1 978343 IC50 = 500000 nM T86702 CXA17I 978344 IC50 = 500000 nM T86702 CXNA13 1201165 IC50 = 14200 nM T86702 CH82ZT 1201321 IC50 = 4190 nM T86702 CAM10Y 1204907 IC50 = 77430 nM T86702 C9IFC6 1348435 IC50 = 110000 nM T86702 C6UZ1A 1383990 IC50 = 58500 nM T86702 CQH3A5 1549481 IC50 > 500000 nM T86702 CN9C8D 2140735 IC50 = 850000 nM T86702 CN6E3U 2366268 IC50 > 10000 nM T86702 CN62WX 2800809 IC50 > 10000 nM T86702 CK3OX7 2916953 IC50 = 47000 nM T86702 CME24U 3649035 IC50 > 101000 nM T86702 C3EI6T 4085085 IC50 = 110000 nM T86702 CC5O4E 4369384 IC50 = 1400 nM T86702 CP8D7Y 4478236 IC50 = 4090 nM T86702 C74PGQ 4907629 IC50 > 2000000 nM T86702 C56JLR 4962547 IC50 = 289000 nM T86702 CQ4VL5 5287415 IC50 = 16 nM T86702 CJ3QI1 5288814 IC50 > 10000 nM T86702 C5IDT0 5289314 Ki = 4500 nM T86702 CO58XD 5311161 IC50 > 100000 nM T86702 CVLS16 5319161 IC50 = 10360 nM T86702 CZC3I7 5326979 IC50 = 200000 nM T86702 CL89FO 5496920 Ki = 127 nM T86702 C1CM3J 6005649 IC50 = 17500 nM T86702 C9S1VI 6006930 IC50 = 48400 nM T86702 CJG2B7 6476333 IC50 = 91410 nM T86702 CL5DH0 6479915 IC50 = 28260 nM T86702 CQEF36 6539670 IC50 = 4 nM T86702 CN5L2B 6852147 Ki = 40 nM T86702 CP2XK7 6882342 IC50 = 230000 nM T86702 CZNK47 6992459 IC50 > 500000 nM T86702 C9Q4MX 7016043 IC50 > 500000 nM T86702 CU3Y1K 7017963 Ki = 28000 nM T86702 C7Y1BX 9543420 IC50 = 24.4 nM T86702 CIJ25V 9794947 IC50 = 90000 nM T86702 C7NP9Z 9798247 IC50 = 1380 nM T86702 CET56A 9801414 Ki = 500 nM T86702 C68HMJ 9801786 IC50 > 10000 nM T86702 CZ6EA7 9802097 IC50 = 640 nM T86702 C4CN0H 9802436 Ki = 0.35 nM T86702 CIXD67 9802768 IC50 = 13 nM T86702 CUSD58 9803469 IC50 = 22100 nM T86702 C4A0XM 9804305 IC50 = 2 nM T86702 C1HP7E 9805710 IC50 = 4.3 nM T86702 CASW18 9806452 Ki = 10 nM T86702 CTK6J8 9808181 IC50 = 23 nM T86702 C5CE8A 9809470 IC50 = 3.7 nM T86702 CTO36D 9817594 IC50 > 100000 nM T86702 C5OE1B 9821883 Ki = 34 nM T86702 C6KJ9W 9822461 IC50 = 28 nM T86702 C6IX7G 9822926 IC50 = 18.1 nM T86702 C1MPW9 9823182 IC50 = 930 nM T86702 CVN5Z3 9823395 IC50 = 1220 nM T86702 C1PW5U 9824010 IC50 = 4 nM T86702 CDJB86 9825720 IC50 = 3.2 nM T86702 CL0G8K 9825927 IC50 = 398.11 nM T86702 C1I6KQ 9826286 Ki = 240 nM T86702 CL59JS 9827846 IC50 = 31 nM T86702 CC1NG5 9829581 IC50 = 29 nM T86702 C7SRM4 9837496 IC50 = 3000 nM T86702 CMAV56 9839147 IC50 = 15 nM T86702 CKF84D 9840581 IC50 = 470 nM T86702 C32JRZ 9843079 Ki = 94 nM T86702 C4RNT6 9845430 IC50 = 1040 nM T86702 CE9AL3 9847113 IC50 = 35 nM T86702 C8IMT2 9847787 IC50 = 2.3 nM T86702 C7VXJ5 9848025 IC50 = 2.7 nM T86702 C4IEK0 9850035 IC50 = 23.9 nM T86702 CD1KW6 9851858 Ki = 2.75 nM T86702 C5DGI9 9851911 IC50 = 1600 nM T86702 C2FYO3 9852206 Ki = 1.73 nM T86702 C7UP3K 9857957 IC50 = 3400 nM T86702 C5TUJ7 9862317 IC50 = 700 nM T86702 C8CEJ4 9862349 IC50 = 480 nM T86702 CS5JT6 9864502 IC50 = 940 nM T86702 CQ0J1G 9865191 IC50 = 3 nM T86702 CI8Z0R 9866250 IC50 = 16 nM T86702 CQ9SG1 9866486 IC50 = 31 nM T86702 C0YN1X 9867935 IC50 = 1320 nM T86702 CJS23I 9868333 Ki = 82 nM T86702 CLQ29X 9869597 IC50 = 1 nM T86702 CG17NZ 9869811 IC50 = 42 nM T86702 C38BVX 9870100 IC50 > 1000 nM T86702 CZO2I0 9870133 IC50 = 100 nM T86702 CA48SX 9870269 IC50 = 5.2 nM T86702 CSM16R 9871355 IC50 = 14600 nM T86702 CHU9I8 9871883 IC50 = 22 nM T86702 C5NM6P 9872886 Ki = 20 nM T86702 CW8IC4 9882151 IC50 > 100000 nM T86702 C0ZT7A 9883002 Ki = 15000 nM T86702 CZBK85 9886177 IC50 = 2000 nM T86702 C4PB5Z 9887544 IC50 = 7.8 nM T86702 C3ZG6O 9887870 Ki = 4.4 nM T86702 CVP45O 9888530 IC50 = 8900 nM T86702 CDW1O4 9888922 IC50 = 3 nM T86702 CD1U5P 9889190 IC50 = 2280 nM T86702 C6TV1K 9889336 IC50 = 5 nM T86702 C27HMG 9889517 IC50 = 1.2 nM T86702 C26SZX 9890226 IC50 = 1.1 nM T86702 CD79UJ 9890632 IC50 = 76000 nM T86702 CU65HY 9891358 IC50 = 10 nM T86702 CO68SM 9891580 IC50 = 62 nM T86702 C3QSE6 9891814 IC50 = 3.3 nM T86702 CF1X0W 9892321 IC50 = 1 nM T86702 CH69LT 9892815 IC50 = 29 nM T86702 CZU7Y4 9892876 IC50 = 45 nM T86702 CX5G0F 9894469 IC50 = 12.88 nM T86702 CSIB97 9896504 IC50 > 30000 nM T86702 C2R5CX 9905493 IC50 = 7 nM T86702 CMSC52 9908418 Ki > 650 nM T86702 CN6WJ1 9909994 IC50 = 570 nM T86702 CJ3K1I 9910075 IC50 = 4560 nM T86702 CM2F7R 9910302 IC50 = 1.7 nM T86702 C6NUE9 9910550 IC50 = 5 nM T86702 CP4LS8 9910727 IC50 = 16300 nM T86702 C62VZI 9912382 IC50 = 0.7 nM T86702 CR98KH 9913488 IC50 = 3 nM T86702 CSZV76 9913881 IC50 = 157 nM T86702 C7ZY1L 9914029 IC50 = 60 nM T86702 C8L2IQ 9915804 Ki = 14 nM T86702 CA3FW0 9918908 IC50 = 0.007 nM T86702 CG1A6B 9924640 IC50 = 28000 nM T86702 C4YGT6 9928325 IC50 = 1.9 nM T86702 C7EIX4 9930068 Ki = 24.1 nM T86702 CK5OV9 9930210 IC50 = 82 nM T86702 CWN0L8 9930514 IC50 = 1750 nM T86702 CCHZ97 9932731 IC50 = 9100 nM T86702 CDXR37 9933197 IC50 = 22 nM T86702 CX17KQ 9933408 IC50 = 5440 nM T86702 C5E7PR 9933720 Ki = 15 nM T86702 C57WSD 9934240 IC50 = 23 nM T86702 C65ION 9935032 IC50 = 76.8 nM T86702 CGFD83 9936194 IC50 = 0.4 nM T86702 C1HRU9 9936228 IC50 = 90 nM T86702 C9OUC8 9936681 IC50 = 0.3 nM T86702 CG38KL 9936728 Ki = 7.8 nM T86702 CE59TP 9936926 IC50 > 10000 nM T86702 CLM2R8 9941370 Ki = 18 nM T86702 C0IBF2 9941371 Ki = 7.31 nM T86702 CY68GC 9945318 IC50 = 30 nM T86702 CB9AO0 9949549 IC50 = 378 nM T86702 C8RXN6 9954304 IC50 > 10000 nM T86702 C32HAZ 9954953 Ki = 28 nM T86702 CK9HX0 9955125 IC50 = 0.2 nM T86702 C8M2RB 9956613 IC50 > 10000 nM T86702 C3Q2UJ 9956686 IC50 = 20 nM T86702 CI5TW9 9956699 IC50 = 1 nM T86702 CC4WG3 9957228 Ki > 300000 nM T86702 CN76XI 9957653 IC50 = 55 nM T86702 CVG0O2 9959014 IC50 > 1000 nM T86702 CN8TK0 9959428 IC50 > 10000 nM T86702 CFQ15E 9976696 IC50 = 16 nM T86702 C0HL2X 9976697 IC50 = 0.7 nM T86702 C09LSY 9979489 Ki > 4501 nM T86702 CXS48O 9979594 Ki = 17 nM T86702 CUA65C 9982414 IC50 = 55 nM T86702 CO09PN 9983251 IC50 = 23 nM T86702 CJGR30 9983604 IC50 = 56.4 nM T86702 CILK24 9983687 Ki = 472 nM T86702 C1N0MZ 9985145 Ki < 2 nM T86702 C8IL6Q 9986000 IC50 = 216 nM T86702 CB2J3S 9999667 IC50 = 80 nM T86702 CO7Y9J 10001450 Ki = 6 nM T86702 C5HN3L 10001964 IC50 = 5 nM T86702 C2L3EU 10003206 Ki = 65 nM T86702 C8Q9OC 10003866 Ki = 11 nM T86702 CVUE46 10005340 Ki = 2 nM T86702 C6U3CK 10006134 IC50 = 6.3 nM T86702 CA8C6U 10008733 Ki = 2.98 nM T86702 C8Q3YW 10008805 IC50 = 400 nM T86702 CR7T3J 10009978 Ki = 582 nM T86702 CJ6H8O 10019658 IC50 = 15 nM T86702 C6WHU4 10023722 IC50 = 280 nM T86702 C71YGT 10025307 Ki = 1300 nM T86702 CM52RO 10030422 IC50 = 1600 nM T86702 CJR59P 10031295 Ki > 4501 nM T86702 CVG03H 10031524 IC50 = 1370 nM T86702 CW74KV 10032055 IC50 = 50 nM T86702 C7J9ZF 10039403 IC50 = 47 nM T86702 CPZ4L1 10041481 IC50 = 500 nM T86702 CW2MK1 10043732 Ki = 10000 nM T86702 CY1J5S 10045091 IC50 = 3800 nM T86702 C7CT4E 10045150 IC50 = 48 nM T86702 CHF92V 10047100 Ki = 3200 nM T86702 CLXN48 10047373 IC50 = 7 nM T86702 CCF5Z4 10047585 IC50 = 0.6 nM T86702 CAN59F 10047708 IC50 = 4 nM T86702 CCA67I 10048718 Ki = 41 nM T86702 CV59KC 10049292 Ki = 570 nM T86702 CZR4U6 10050655 Ki = 62 nM T86702 C19LUE 10050937 Ki = 6 nM T86702 CLZ87W 10051236 Ki = 2105 nM T86702 C1G0HE 10051959 IC50 = 2976 nM T86702 CZ6R1T 10052198 Ki = 12 nM T86702 CSHD67 10054852 IC50 = 1.1 nM T86702 CD3RL7 10070821 Ki > 10000 nM T86702 C2P7WT 10070826 Ki = 54 nM T86702 CQ7PJ9 10072419 Ki = 12 nM T86702 CB28NP 10073353 IC50 = 10000 nM T86702 CSG9A5 10073761 Ki = 14 nM T86702 CJK0R1 10074190 IC50 = 98 nM T86702 CV0I9M 10074738 IC50 = 1523 nM T86702 CJ2H0T 10077849 IC50 = 121 nM T86702 CUT28D 10088847 Ki = 69.8 nM T86702 C8AEK4 10093420 IC50 = 1.2 nM T86702 C5W4ZA 10094362 IC50 = 400 nM T86702 CHK0M7 10094867 Ki = 112 nM T86702 CA6X2Z 10095338 IC50 = 7.8 nM T86702 CMY3X2 10098158 IC50 = 5.1 nM T86702 C2XV5J 10098250 IC50 = 40.6 nM T86702 CLF2R6 10098574 Ki = 6 nM T86702 C3V2HW 10099112 IC50 = 7 nM T86702 CMLA47 10099961 IC50 = 2169 nM T86702 CF3HQ9 10100283 Ki < 2 nM T86702 CU3X8V 10115845 IC50 = 3700 nM T86702 CGW13V 10116395 IC50 = 400 nM T86702 C7A8MI 10120093 IC50 = 42.5 nM T86702 CP65KL 10125869 Ki = 300 nM T86702 CYU19P 10127901 Ki > 4500 nM T86702 CH0UW2 10129190 Ki > 4500 nM T86702 C6MSI0 10141443 IC50 = 6000 nM T86702 CD3U8E 10150649 Ki = 11 nM T86702 CUG62E 10155007 IC50 > 40000 nM T86702 CLQ89T 10155008 IC50 > 40000 nM T86702 CR5H6E 10163627 Ki = 2609 nM T86702 CZO5V4 10164317 IC50 = 13.8 nM T86702 CNTC03 10172417 Ki = 7.7 nM T86702 CGB27E 10174981 Ki > 4500 nM T86702 CL47AR 10175070 Ki > 4500 nM T86702 C4ULO6 10175077 Ki > 4500 nM T86702 C84ZQD 10175219 Ki > 4500 nM T86702 CIT0H4 10175323 Ki > 4500 nM T86702 C95IGP 10175331 Ki > 4500 nM T86702 CT7U0M 10175426 Ki > 4500 nM T86702 CGMU01 10183812 IC50 = 62 nM T86702 CYV78C 10184127 IC50 = 460 nM T86702 CK0P3F 10186536 Ki > 4501 nM T86702 C51RPY 10195069 Ki > 4500 nM T86702 CCHX74 10195307 Ki > 4500 nM T86702 C94KHT 10195527 Ki > 4500 nM T86702 CDG35O 10196192 Ki = 3690 nM T86702 CVRZ27 10198038 IC50 > 100000 nM T86702 C4K1MJ 10208262 Ki = 3915 nM T86702 CG8FA4 10218128 Ki > 4500 nM T86702 C7Y2US 10218353 Ki > 4500 nM T86702 CV5X8A 10224181 IC50 > 30000 nM T86702 C06HYC 10227441 IC50 = 10000 nM T86702 C7T0WH 10229644 IC50 = 221 nM T86702 CCRM18 10231253 IC50 = 2.2 nM T86702 CO8M7Q 10239526 Ki > 4500 nM T86702 CEO4X5 10239762 Ki > 4500 nM T86702 CU7TQ3 10239803 Ki > 4500 nM T86702 CQ1E4F 10248274 Ki = 2187.76 nM T86702 CLAX20 10250594 IC50 = 25 nM T86702 C0J3TC 10250722 Ki = 600 nM T86702 CHGB94 10251825 Ki = 38 nM T86702 CBM0Y4 10252411 Ki < 100 nM T86702 CLX62O 10252774 Ki = 9 nM T86702 CK9DF5 10253223 IC50 = 27000 nM T86702 C2V4MP 10253549 IC50 = 4.295 nM T86702 CQF3V9 10253673 IC50 = 4360 nM T86702 CD8QY2 10253933 IC50 > 10000 nM T86702 CJ3Q8W 10256080 IC50 = 1485 nM T86702 CB6SE4 10256227 IC50 = 110 nM T86702 CO47KX 10256290 Ki = 5 nM T86702 C8OUE9 10256513 Ki = 5 nM T86702 C4WV7B 10257654 IC50 = 481 nM T86702 C0CE3N 10269452 IC50 > 40000 nM T86702 C0QS9V 10269453 IC50 = 2300 nM T86702 C2MES9 10271604 IC50 = 91000 nM T86702 CH68BK 10273973 IC50 = 450 nM T86702 C3IG0K 10280852 IC50 = 115 nM T86702 CR48SA 10289842 Ki > 4500 nM T86702 CO60CU 10290029 Ki > 4500 nM T86702 CJ9WI1 10296950 IC50 = 1500 nM T86702 C1HK6G 10299554 IC50 = 670 nM T86702 C2JAZ9 10301436 IC50 = 690 nM T86702 CE1KM9 10311498 Ki > 4500 nM T86702 CJ15OB 10311501 Ki > 4500 nM T86702 C5F0EV 10311947 Ki > 4500 nM T86702 C7G6QW 10312268 Ki > 4500 nM T86702 CQ5IT9 10312372 Ki > 4500 nM T86702 C37ZDM 10317565 Ki > 10000 nM T86702 C2U6MY 10318916 Ki = 3.7 nM T86702 CIDW49 10319098 Ki > 4501 nM T86702 CG23FV 10320328 IC50 = 5 nM T86702 CJWH74 10321975 Ki > 4501 nM T86702 CFQ4U0 10322451 Ki = 19 nM T86702 CY08WJ 10322755 Ki = 762 nM T86702 C50KSE 10323483 IC50 = 82 nM T86702 C9DR2I 10323789 IC50 = 309 nM T86702 CQH5D4 10324032 IC50 = 1.5 nM T86702 CPI8R0 10324532 Ki = 33 nM T86702 C1C4VZ 10326004 Ki = 384 nM T86702 CF5UN8 10326272 IC50 = 1400 nM T86702 C5F0RK 10326931 IC50 = 314 nM T86702 CG6NT9 10338869 IC50 = 2600 nM T86702 C0W6IH 10339389 IC50 = 600 nM T86702 C7UZA4 10340758 IC50 = 9.6 nM T86702 CCK1A4 10342176 IC50 = 24000 nM T86702 CFO74N 10343375 Ki = 4000 nM T86702 CJIW74 10343996 IC50 = 14 nM T86702 CW1VL2 10345348 IC50 = 12500 nM T86702 CPJ1G8 10345717 IC50 = 5633 nM T86702 CX8H3Z 10346437 IC50 > 10000 nM T86702 C94ANQ 10347529 IC50 = 26 nM T86702 C9GV5Z 10348475 IC50 = 120 nM T86702 CNP78B 10348836 Ki = 9.5 nM T86702 C50DNH 10362338 Ki = 426.58 nM T86702 C9FU5G 10362663 IC50 = 1.3 nM T86702 CL4B2U 10364155 IC50 > 10000 nM T86702 CH89GT 10365752 IC50 = 4.5 nM T86702 CI0T8K 10366352 Ki > 4501 nM T86702 C6FJU3 10367981 IC50 > 10000 nM T86702 C8DJX4 10368307 Ki = 38 nM T86702 CJ96GA 10370197 IC50 = 178 nM T86702 C5VHS0 10370227 IC50 = 2340 nM T86702 C6T4WO 10370281 Ki = 373 nM T86702 CDY02J 10370532 Ki = 21 nM T86702 C5X3AI 10380124 IC50 = 600 nM T86702 CEM0U7 10387692 IC50 > 10000 nM T86702 CL97HT 10388523 Ki = 29.6 nM T86702 CZNT94 10389113 IC50 = 100 nM T86702 CP9WG5 10389610 IC50 = 38 nM T86702 CB6IH4 10389682 Ki = 16 nM T86702 CR38WZ 10392467 IC50 = 1303 nM T86702 C8UTS7 10393307 IC50 = 518 nM T86702 C16BSA 10394828 IC50 = 50000 nM T86702 CFKA79 10395015 Ki > 2000 nM T86702 C9HM1A 10402302 IC50 = 620000 nM T86702 CLP05D 10407603 IC50 = 3.4 nM T86702 CTX2S3 10410319 Ki = 25 nM T86702 CRD6Z4 10410935 IC50 > 10000 nM T86702 CZ90OC 10412486 Ki = 3 nM T86702 CA0TY8 10413076 Ki = 265 nM T86702 C98HMP 10413940 Ki = 2400 nM T86702 CJ95UZ 10414150 IC50 = 1159 nM T86702 CH1S2G 10414974 Ki = 277 nM T86702 CV4JT6 10415842 IC50 = 295 nM T86702 C4J7IP 10416507 Ki = 8 nM T86702 CZ3D4T 10428502 IC50 = 16 nM T86702 C0V9FN 10433382 IC50 = 4.365 nM T86702 CS32HR 10435935 IC50 = 3.4 nM T86702 CO6VM2 10436776 IC50 = 5970 nM T86702 C7XE1L 10437629 IC50 = 1500 nM T86702 C9QS8N 10438212 IC50 = 427 nM T86702 C5WV1N 10439082 Ki > 2000 nM T86702 CA75GC 10453674 IC50 > 10000 nM T86702 C54UDR 10453826 IC50 = 200 nM T86702 CP9WB1 10454818 Ki = 360 nM T86702 CA5W6I 10458439 IC50 = 1895 nM T86702 CP13CG 10459563 IC50 = 2194 nM T86702 CA7DM9 10474389 IC50 = 100 nM T86702 CWV9Q2 10477531 Ki = 6.67 nM T86702 CP30UC 10478059 Ki = 700 nM T86702 C87WDS 10478481 Ki = 42.66 nM T86702 CHG02V 10478612 Ki = 6.75 nM T86702 C9VIP5 10479752 Ki = 91.2 nM T86702 CHL30D 10482442 IC50 = 2473 nM T86702 CNQZ36 10483139 Ki = 28 nM T86702 COE94R 10484032 IC50 = 50 nM T86702 C3UT8Z 10492262 IC50 = 29000 nM T86702 COT6G1 10492779 Ki = 30902.95 nM T86702 CO92UA 10494668 Ki = 16982.44 nM T86702 C9KHT4 10495552 Ki = 404 nM T86702 CV8U1L 10497756 IC50 = 49300 nM T86702 C6KD0A 10498747 IC50 = 0.7 nM T86702 C9YIS7 10501217 IC50 = 20 nM T86702 CK4E0P 10501888 Ki = 510 nM T86702 CZ2UY0 10502046 IC50 = 6.6 nM T86702 C36OMW 10502172 IC50 = 57 nM T86702 C1EAW7 10502187 Ki = 810 nM T86702 C5V8HJ 10502382 IC50 < 1 nM T86702 CJZ5T8 10502487 IC50 > 10000 nM T86702 CK12GT 10502537 Ki = 104 nM T86702 CSN17G 10502708 IC50 = 10 nM T86702 CZ1R5Q 10502869 Ki = 13500 nM T86702 CBNM82 10503128 IC50 = 6.3 nM T86702 C9LJR5 10503737 IC50 = 26 nM T86702 C5Y4IA 10504081 IC50 = 10700 nM T86702 CD80YF 10504445 IC50 = 9 nM T86702 C2C7TE 10504472 IC50 = 3 nM T86702 CK2AB5 10505370 Ki = 1500 nM T86702 CV19QD 10505495 Ki = 1000 nM T86702 CH6S8Y 10505729 IC50 > 10000 nM T86702 C6D7JF 10506147 IC50 = 22 nM T86702 C7S0DB 10506158 IC50 = 3520 nM T86702 CS8V1G 10507004 Ki = 52 nM T86702 CV2T7C 10507137 Ki = 350 nM T86702 CFJ96A 10507282 Ki = 39 nM T86702 C9C5EL 10521197 IC50 = 2.3 nM T86702 CBT12Q 10522080 IC50 = 15 nM T86702 CC2F5Y 10522311 IC50 = 18 nM T86702 CZ36JW 10523383 IC50 = 135 nM T86702 CQEH42 10524134 IC50 = 9 nM T86702 CYU87N 10524260 IC50 = 15 nM T86702 C79NQP 10524926 Ki = 60.26 nM T86702 COT07L 10525329 IC50 = 74.99 nM T86702 C61GSD 10525562 IC50 = 7.5 nM T86702 C14XUW 10526101 IC50 = 66 nM T86702 CU4H1A 10526209 Ki = 42 nM T86702 CJK6G1 10526509 IC50 = 12 nM T86702 CWLD37 10526788 IC50 = 23 nM T86702 CA0J2K 10527557 Ki = 81 nM T86702 CHS9Q5 10527785 IC50 = 22 nM T86702 C2H8XM 10527787 Ki = 65 nM T86702 CJ0D7G 10528505 IC50 = 3.2 nM T86702 CYGU41 10529315 IC50 = 4560 nM T86702 CIOJ69 10529720 Ki = 200 nM T86702 C6PGE1 10530040 Ki = 49 nM T86702 C30UCT 10530499 Ki = 5 nM T86702 CEV6I5 10531005 Ki = 40 nM T86702 CJ2TZ3 10531167 Ki = 21 nM T86702 CS0AD8 10532048 Ki = 10 nM T86702 C86EWV 10541018 IC50 = 130500 nM T86702 CS2MR3 10542854 IC50 > 1000000 nM T86702 CJ8D5M 10542855 IC50 = 34000 nM T86702 CGE54K 10543918 Ki = 4073.8 nM T86702 CB7TX1 10543975 Ki = 3200 nM T86702 CO2R0P 10544323 IC50 = 269 nM T86702 CQJA07 10544993 Ki = 290 nM T86702 CJ57BA 10545870 Ki = 113 nM T86702 C1VZ0D 10546808 Ki = 1300 nM T86702 C4PK0U 10549114 IC50 = 7.2 nM T86702 C4TA1K 10549256 IC50 = 2 nM T86702 CHCI01 10549577 IC50 = 9 nM T86702 C2HJ1U 10549764 IC50 = 60 nM T86702 CRHP20 10550304 IC50 = 27 nM T86702 C7WQ5Z 10550399 IC50 = 5 nM T86702 CNQ75F 10551139 IC50 = 172.98 nM T86702 CCH0K3 10551483 IC50 = 9.499 nM T86702 CWF2H8 10551771 IC50 = 300 nM T86702 C5UD0A 10551910 IC50 = 20 nM T86702 C8VUQ4 10552056 Ki = 50 nM T86702 CNE73L 10552476 IC50 = 10.99 nM T86702 COYU34 10553872 Ki = 95 nM T86702 C0S6GT 10554037 Ki = 15 nM T86702 CSQC42 10554611 Ki = 19 nM T86702 C7P5AW 10554727 Ki = 49 nM T86702 CI8XG0 10554869 IC50 = 21 nM T86702 CYJ41F 10554927 Ki = 1100 nM T86702 CWJ48L 10569469 Ki = 336 nM T86702 CT7O9M 10569678 IC50 = 3 nM T86702 C8RWE4 10569743 IC50 = 36 nM T86702 CE14GM 10570702 IC50 = 8 nM T86702 CE7G5A 10570770 Ki = 66 nM T86702 C2MD1V 10571436 IC50 = 9170 nM T86702 CBXZ79 10572150 IC50 = 14 nM T86702 CPF0R5 10572544 Ki = 700 nM T86702 CYX52N 10572651 Ki = 930 nM T86702 C21VZS 10573362 IC50 = 100 nM T86702 CS9Y3Q 10573446 IC50 = 6 nM T86702 C61IUN 10574937 IC50 = 45 nM T86702 CK3JV9 10576740 IC50 = 18 nM T86702 CJ7KH8 10578213 Ki = 12 nM T86702 C1KH7E 10578728 IC50 = 2850 nM T86702 C9L5OM 10579282 IC50 = 19.5 nM T86702 CI0E7L 10587235 IC50 = 310 nM T86702 CIUO27 10593253 IC50 = 16 nM T86702 CJSX87 10593373 Ki = 305 nM T86702 CB20LM 10594000 Ki = 70 nM T86702 CUTS47 10594564 IC50 = 6 nM T86702 CN4Y6H 10594565 IC50 = 5 nM T86702 CD65OG 10594830 IC50 = 407.38 nM T86702 CT8Z2B 10594938 Ki = 36 nM T86702 CUN73L 10595134 Ki = 1995.26 nM T86702 CYNC76 10596158 IC50 = 12 nM T86702 C6M1HR 10599498 Ki = 44 nM T86702 C0R8ND 10599533 IC50 = 7 nM T86702 CQCW86 10599579 IC50 = 5 nM T86702 CW18QK 10599594 IC50 = 2.692 nM T86702 CR1JI4 10600645 IC50 = 12 nM T86702 C5WUG1 10601082 Ki = 1400 nM T86702 C6RH4O 10601640 IC50 = 174.98 nM T86702 C84URB 10610500 Ki = 165958.69 nM T86702 CE2QR9 10613211 Ki = 1760 nM T86702 CZD9B3 10617580 IC50 = 4.3 nM T86702 CC1T5D 10618255 Ki = 61 nM T86702 CL02BO 10618584 IC50 = 8 nM T86702 CM06XN 10620633 IC50 = 10300 nM T86702 C8IZN2 10620836 IC50 = 2400 nM T86702 CZL9Y4 10621353 Ki = 700 nM T86702 C0JGS3 10621776 IC50 = 30 nM T86702 CL5QN9 10622296 IC50 = 15 nM T86702 CL62YC 10622822 IC50 = 87.1 nM T86702 CZJB31 10622970 IC50 = 54 nM T86702 CL67UQ 10623250 IC50 = 9000 nM T86702 CQH75Y 10624313 Ki = 490 nM T86702 CGB29T 10625771 IC50 = 12 nM T86702 C98KGO 10625860 IC50 = 385.48 nM T86702 C6H9CT 10626366 Ki = 2000 nM T86702 C3NKC0 10626927 Ki = 11 nM T86702 CL43CO 10627365 IC50 = 22 nM T86702 CM1F5B 10636628 Ki = 69000 nM T86702 C54TIA 10640100 Ki = 4365.16 nM T86702 CE8WK2 10640178 Ki = 94 nM T86702 C7KGM3 10642071 IC50 = 16 nM T86702 CWRY91 10642128 IC50 = 20 nM T86702 CXS86T 10642533 Ki = 141 nM T86702 CI2QB9 10642965 IC50 = 2 nM T86702 CU5D3S 10645086 Ki = 46 nM T86702 C13BAC 10645799 Ki = 28 nM T86702 C2O1XM 10647817 IC50 = 13 nM T86702 C4TXZ1 10648776 Ki = 580 nM T86702 C5RWF4 10648802 IC50 = 2.5 nM T86702 CX48UV 10649092 IC50 = 6 nM T86702 C6S1KA 10649216 IC50 > 10000 nM T86702 C0A5XB 10658473 IC50 = 99000 nM T86702 C27QHB 10663143 IC50 = 48 nM T86702 CGSX70 10664302 IC50 = 67.9 nM T86702 C97KZU 10665624 IC50 = 10 nM T86702 C49AZV 10665669 IC50 = 20 nM T86702 C4A0WY 10667012 Ki = 77.62 nM T86702 CF0E6H 10668745 IC50 = 9 nM T86702 C4HJS1 10669027 Ki = 1000 nM T86702 C8HK0C 10669534 IC50 = 60 nM T86702 CAI72H 10670246 IC50 = 14 nM T86702 C3B8KZ 10670761 Ki = 151 nM T86702 CY6QC1 10670819 IC50 = 114 nM T86702 CPG5O2 10671155 IC50 = 16.98 nM T86702 C09LJR 10671827 IC50 = 41 nM T86702 C17LYV 10672346 IC50 = 2428 nM T86702 CMU74I 10672857 IC50 = 8620 nM T86702 CU6Y4O 10674458 Ki = 1500 nM T86702 C9OIB3 10686890 Ki = 1820 nM T86702 CBO26H 10687032 IC50 = 175 nM T86702 CXTP56 10688727 IC50 = 3 nM T86702 C0OJ9C 10689683 IC50 = 87 nM T86702 CR3Q8Z 10691191 Ki = 104 nM T86702 CSA80H 10692194 IC50 = 8 nM T86702 CS5CL7 10692307 IC50 = 2 nM T86702 C4Q1XY 10692726 Ki = 39 nM T86702 CR5KF8 10692994 IC50 = 290 nM T86702 CDI12G 10693559 IC50 = 10 nM T86702 CB70DA 10693592 IC50 = 12 nM T86702 C8IG5Q 10693625 Ki = 31 nM T86702 CVML68 10693881 IC50 = 2 nM T86702 CZGC63 10695865 IC50 = 5060 nM T86702 CVQF97 10695971 IC50 = 7 nM T86702 CW6CF7 10696226 IC50 = 6 nM T86702 C6MWX8 10696713 IC50 = 410.02 nM T86702 C1YFC3 10696977 IC50 = 3920 nM T86702 C4BME8 10697140 IC50 = 1810 nM T86702 CBN9K8 10697378 Ki = 11 nM T86702 C1O5CQ 10697393 Ki = 74 nM T86702 CM4AI6 10698165 Ki = 12 nM T86702 C4THQ9 10698311 Ki = 27 nM T86702 C6Y1OU 10698367 Ki = 4 nM T86702 C14TWR 10708950 IC50 = 694000 nM T86702 CKQ6N5 10708951 Ki = 16000 nM T86702 CJXO26 10709434 Ki = 5000 nM T86702 C7CI4T 10713194 Ki = 100 nM T86702 CJZ0X3 10714009 Ki = 460 nM T86702 CG38ZD 10714323 IC50 = 300 nM T86702 C2GL3A 10714610 Ki = 600 nM T86702 C09ZXY 10714796 Ki = 70 nM T86702 C4IWF2 10714988 IC50 = 48 nM T86702 CO9KV7 10715115 IC50 = 1 nM T86702 CE1D6G 10716217 IC50 = 0.7 nM T86702 CF98LK 10716463 Ki = 380 nM T86702 CF51EI 10716486 IC50 = 146.99 nM T86702 C0ZX6T 10717308 IC50 = 7 nM T86702 C7OSW8 10718200 IC50 = 8 nM T86702 CI64YZ 10718883 IC50 = 27 nM T86702 C35MRE 10719092 IC50 = 5 nM T86702 CVW81M 10719595 IC50 = 6600 nM T86702 C4RD0P 10719602 Ki = 860 nM T86702 CI96XV 10720740 Ki = 9 nM T86702 CIV3P5 10720775 Ki = 65 nM T86702 C65IGZ 10720864 Ki = 13 nM T86702 CTGL64 10721152 Ki = 690 nM T86702 C4J1WN 10721454 IC50 = 10 nM T86702 CG4DA0 10731747 IC50 = 2550 nM T86702 CU91MQ 10732988 Ki = 3235.94 nM T86702 C37LUZ 10734191 Ki = 2500 nM T86702 C0TI1M 10734897 IC50 = 1600 nM T86702 C8KE2C 10735676 IC50 > 20000 nM T86702 CBHX39 10736792 Ki = 400 nM T86702 C51DZG 10737732 IC50 = 9 nM T86702 CA28EM 10738103 Ki = 236 nM T86702 C1LS5U 10738104 IC50 = 5 nM T86702 CL74TG 10738165 IC50 = 14 nM T86702 C2W0RV 10738429 Ki = 125 nM T86702 CQ7HY1 10738924 Ki = 63 nM T86702 CLME42 10739270 Ki = 100 nM T86702 C76ANK 10739335 IC50 = 3.499 nM T86702 C0T2VK 10740460 IC50 = 39 nM T86702 CKJD45 10741133 IC50 = 810 nM T86702 CL64BU 10741592 IC50 = 10.96 nM T86702 C4MQ8L 10742072 IC50 = 8 nM T86702 CKX5R3 10742142 IC50 = 777 nM T86702 CPA73X 10742152 Ki = 69 nM T86702 CHW23E 10742387 IC50 = 89.13 nM T86702 CCH94Q 10743507 IC50 = 13 nM T86702 C1LF0S 10744337 Ki = 21 nM T86702 CEV8X0 10744751 Ki = 13 nM T86702 CSM9H7 10745124 Ki = 120 nM T86702 C9ILP3 10745718 IC50 = 28 nM T86702 C4IF2L 10745725 Ki = 2 nM T86702 C3CEX9 10755223 Ki = 7000 nM T86702 CMZC64 10756622 IC50 = 258 nM T86702 CE09PI 10757715 IC50 = 23 nM T86702 CTKR07 10758266 Ki = 3300 nM T86702 C03KYQ 10760373 Ki = 90 nM T86702 CF7SH1 10761128 IC50 = 20 nM T86702 CLEG16 10761206 Ki = 200 nM T86702 C0BAE9 10763583 IC50 = 15400 nM T86702 C68THN 10763851 IC50 = 5 nM T86702 CM54WS 10764477 Ki = 35000 nM T86702 CAG53Y 10764489 IC50 = 16.98 nM T86702 C7X6EC 10764497 Ki = 3800 nM T86702 C0ZJB9 10764600 IC50 = 184.08 nM T86702 CJE76M 10764871 IC50 = 12 nM T86702 CQ0KM4 10765140 IC50 = 5 nM T86702 CXOL83 10765385 Ki = 48 nM T86702 CD58QP 10765874 IC50 = 2000 nM T86702 C3P2TS 10766036 IC50 = 3330 nM T86702 CJW2B7 10766518 IC50 = 60 nM T86702 CN6P1J 10766950 IC50 = 10 nM T86702 CWR5Z3 10767105 IC50 > 9999 nM T86702 CR4I1E 10767157 IC50 = 3570 nM T86702 C7Q2EM 10767236 IC50 = 36 nM T86702 CNT4D0 10767387 Ki = 93 nM T86702 C1M8BZ 10767542 IC50 = 400 nM T86702 C18QVD 10768090 Ki = 11 nM T86702 CQ7J4I 10769007 IC50 = 17400 nM T86702 C6VKJ9 10769394 Ki = 1400 nM T86702 CIN4A9 10783989 Ki = 300 nM T86702 C0QW3C 10784639 Ki = 57.54 nM T86702 CH3MK8 10785400 Ki = 38 nM T86702 C31KWI 10785840 Ki = 660 nM T86702 CLAP90 10785969 IC50 > 1000 nM T86702 CGE9V4 10787514 Ki = 23 nM T86702 C2FA7J 10787997 IC50 = 8 nM T86702 C16XQR 10788211 IC50 = 13 nM T86702 C0DFB9 10788617 IC50 = 1.1 nM T86702 CNAE08 10788733 IC50 = 16 nM T86702 CXQD12 10789326 IC50 > 10000 nM T86702 CKV2O8 10789493 IC50 = 5.297 nM T86702 CM74LH 10789594 IC50 > 1000 nM T86702 C45UGJ 10789671 IC50 = 4 nM T86702 C9NZ4W 10789711 IC50 = 8.892 nM T86702 CN6M3W 10789971 Ki = 85 nM T86702 C8EOY6 10790150 Ki = 140 nM T86702 CHWG02 10790787 IC50 = 2340 nM T86702 CF4T1N 10791150 Ki = 270 nM T86702 CWCD73 10805054 IC50 = 14 nM T86702 C1WZ4S 10805349 IC50 = 5.8 nM T86702 CIV42N 10807240 Ki = 1260 nM T86702 C9VML0 10807861 Ki = 2300 nM T86702 C2GMT4 10808023 Ki = 5350 nM T86702 CN8I3Z 10808172 IC50 = 69 nM T86702 CQX5P6 10808260 IC50 = 8 nM T86702 CKV36G 10808884 IC50 = 20 nM T86702 C5HF8Z 10809178 IC50 = 4045 nM T86702 CT1AI4 10810573 IC50 = 42 nM T86702 CV3ZA5 10812444 IC50 = 123.88 nM T86702 CZB7L2 10812929 IC50 = 6.5 nM T86702 C4TF0K 10813874 IC50 = 17 nM T86702 CCIL63 10813879 IC50 = 13 nM T86702 CIUN51 10814028 IC50 = 10100 nM T86702 C80CZA 10815208 IC50 = 1290 nM T86702 CS7BY4 10816934 IC50 = 10 nM T86702 C47NJR 10823585 IC50 > 2000000 nM T86702 CX2E1C 10829071 IC50 = 14 nM T86702 CR0U8Z 10829213 IC50 = 23000 nM T86702 C31LBN 10831751 Ki = 192 nM T86702 C3AI5Z 10831752 IC50 = 17 nM T86702 CLK9P7 10832592 IC50 = 737 nM T86702 CF50HD 10832925 IC50 = 10 nM T86702 CV57JB 10833044 Ki = 1130 nM T86702 C8NCA2 10833242 Ki = 1122.02 nM T86702 C5OG4U 10833497 IC50 = 15 nM T86702 C2A0IX 10833840 IC50 = 17 nM T86702 CH90ZB 10834348 IC50 = 18.5 nM T86702 C9M1JI 10834357 Ki = 92 nM T86702 C2IKW6 10836183 Ki = 107 nM T86702 C48PYQ 10836923 IC50 = 28 nM T86702 CH8OV4 10837276 IC50 = 33 nM T86702 CF40VH 10837557 IC50 = 8 nM T86702 CY4J9A 10838149 IC50 = 10 nM T86702 CHWQ34 10839761 Ki = 1200 nM T86702 CA76MU 10840059 IC50 > 10000 nM T86702 CPD3L7 10840455 Ki = 31 nM T86702 CR2UX3 10840602 Ki = 25 nM T86702 CI0HR4 10840639 Ki = 37 nM T86702 C6PU8A 10840863 Ki = 9400 nM T86702 C0PL9V 10849322 IC50 = 318000 nM T86702 C1ZWH6 10849395 Ki = 16000 nM T86702 CEG8T6 10852576 IC50 = 1040 nM T86702 C9TIR6 10853176 Ki = 933.25 nM T86702 C0W6AK 10854448 Ki = 5248.07 nM T86702 C9EU2B 10854874 Ki = 4073.8 nM T86702 CF72UK 10864417 IC50 = 169 nM T86702 CBQ70P 10874312 IC50 = 6.2 nM T86702 CXY47P 10875332 IC50 = 253 nM T86702 CXGN38 10875470 IC50 = 79 nM T86702 C3AY8O 10885569 IC50 = 103 nM T86702 CAU0I3 10885834 IC50 = 69.6 nM T86702 CA64PN 10886607 IC50 = 84 nM T86702 C0R5QL 10894433 Ki = 5.2 nM T86702 CPJ0I8 10896934 IC50 = 64 nM T86702 CU7YE0 10896986 IC50 = 1.6 nM T86702 CMV89R 10897017 IC50 = 156 nM T86702 CX93MR 10907320 IC50 = 134 nM T86702 CSK87I 10907725 IC50 = 62 nM T86702 C2M4PK 10916140 Ki > 650 nM T86702 CGI2T1 10928606 IC50 = 1.2 nM T86702 CXHA75 10928874 IC50 = 162 nM T86702 CXY4L6 10929354 IC50 = 8 nM T86702 CDSQ41 10929404 IC50 = 62 nM T86702 CWO29J 10940364 IC50 = 474 nM T86702 CL64UM 10940712 IC50 = 49 nM T86702 C2TA9N 10949166 Ki = 5.2 nM T86702 C9YOU4 10951375 IC50 = 15.1 nM T86702 CJI1G0 10951750 IC50 = 1.6 nM T86702 C7PX8G 10960109 Ki > 650 nM T86702 CU2Q8S 10971085 IC50 = 16 nM T86702 CL7K8S 10983560 Ki < 1 nM T86702 CR9J5B 10983887 IC50 = 18 nM T86702 CJ8I9G 10983916 IC50 = 273 nM T86702 C0NIX9 10985227 IC50 = 218 nM T86702 CCX0L6 10994350 IC50 = 5.4 nM T86702 CA5I7L 10995373 IC50 = 76 nM T86702 C4PNK3 11006191 IC50 = 705 nM T86702 C8ERT5 11014626 Ki > 650 nM T86702 C75DGS 11015731 Ki = 617 nM T86702 CG2DK0 11016448 IC50 = 41.8 nM T86702 CF30UR 11016519 IC50 = 5.7 nM T86702 CODQ51 11016616 IC50 = 33.7 nM T86702 CO6C8A 11017232 IC50 = 200 nM T86702 CM1H5P 11026185 Ki = 48 nM T86702 CQD70Y 11026301 Ki > 650 nM T86702 C6IHF5 11026991 IC50 > 100 nM T86702 C0ERN9 11037836 Ki > 650 nM T86702 C83AKP 11038896 IC50 = 122 nM T86702 CG3B5N 11039339 IC50 = 214 nM T86702 CZ0RX5 11048356 Ki = 11000 nM T86702 CZO40T 11048604 Ki > 650 nM T86702 C23KPN 11050468 IC50 = 3.7 nM T86702 CYA27S 11059553 Ki = 2.88 nM T86702 C9RU4I 11059620 IC50 = 657 nM T86702 C1N5PT 11070986 IC50 = 739 nM T86702 C18EIZ 11071831 IC50 = 45.5 nM T86702 C2LSU0 11072397 IC50 = 115 nM T86702 C7VKE3 11080910 Ki = 22.3 nM T86702 CG0A4C 11081333 IC50 = 184 nM T86702 CVJX34 11081788 Ki = 3.4 nM T86702 C05MUK 11081992 IC50 = 4.2 nM T86702 C6XI8J 11082293 IC50 = 31 nM T86702 CF0NJ9 11090097 IC50 = 9 nM T86702 CS29GX 11091928 IC50 = 3 nM T86702 CE8V9B 11092295 IC50 = 10.3 nM T86702 CR8ZA7 11092551 IC50 = 305 nM T86702 CWT6C7 11092884 IC50 = 203 nM T86702 CX69YN 11093502 IC50 = 2.5 nM T86702 C8CK3E 11102531 IC50 = 278 nM T86702 C57OXT 11102540 Ki = 3.33 nM T86702 CA2OS3 11103408 IC50 = 47 nM T86702 CY1SR9 11113744 IC50 = 399 nM T86702 CI1GS5 11114351 IC50 = 1490 nM T86702 CUO7B3 11122933 Ki = 16.2 nM T86702 C8YVE5 11123989 IC50 = 21 nM T86702 C3PR1J 11124862 IC50 = 155 nM T86702 CAJ27B 11124943 IC50 = 17 nM T86702 CNBG53 11124956 IC50 = 4.7 nM T86702 C2YBQ7 11134935 IC50 = 345 nM T86702 C8DMW5 11135133 IC50 = 694 nM T86702 CD3N8B 11135304 IC50 = 195 nM T86702 CT1RP5 11143436 IC50 = 50000 nM T86702 C5WS3E 11147931 IC50 > 100000 nM T86702 CCQ6N8 11194666 IC50 > 100000 nM T86702 C43ONW 11202395 Ki > 4501 nM T86702 CO76XI 11205873 IC50 = 100000 nM T86702 C9R7OM 11207122 IC50 = 30000 nM T86702 CPV9L7 11246575 Ki = 3.3 nM T86702 CUOH67 11252195 IC50 > 100000 nM T86702 CJZ3P6 11257884 Ki = 92 nM T86702 CO7T3M 11261246 IC50 = 130 nM T86702 CP17ID 11284983 IC50 = 144 nM T86702 CF9O2R 11286824 IC50 = 80000 nM T86702 C1IW7N 11292680 IC50 = 50 nM T86702 C8C5AV 11294179 Ki > 10000 nM T86702 CK91YW 11317404 IC50 > 5000 nM T86702 CLH50U 11318841 IC50 = 492 nM T86702 CJ5SU9 11328354 Ki > 300000 nM T86702 CN2P4G 11328571 IC50 > 5000 nM T86702 C0XR3B 11330861 IC50 = 1090 nM T86702 CQH57S 11342435 IC50 = 81 nM T86702 CCKI02 11360440 Ki = 2 nM T86702 C7QNX8 11363138 IC50 > 5000 nM T86702 CM8Y1J 11367571 IC50 > 100000 nM T86702 C48DYJ 11374008 Ki = 2.1 nM T86702 C9ABX8 11397130 Ki > 4501 nM T86702 C13NCF 11400989 IC50 = 50000 nM T86702 C3EX5J 11407165 Ki = 50 nM T86702 CI0V6L 11447356 IC50 > 100000 nM T86702 COS67B 11456566 IC50 = 1060 nM T86702 CCMT46 11457732 IC50 = 90000 nM T86702 CQ1D6E 11470070 IC50 = 1000 nM T86702 C5G8PM 11511807 IC50 > 5000 nM T86702 C5VUM2 11517085 Ki = 7700 nM T86702 C1NZB9 11548265 IC50 = 42.5 nM T86702 CIWP38 11555036 IC50 = 366 nM T86702 CHV2G1 11575995 Ki > 10000000 nM T86702 C3H2DG 11577137 IC50 = 942 nM T86702 CVGC49 11603611 Ki = 5 nM T86702 CUL5H2 11605631 IC50 = 237 nM T86702 CXKU59 11620780 IC50 > 5000 nM T86702 CNY92D 11640694 Ki > 50000 nM T86702 CFV49P 11641262 IC50 < 1.5 nM T86702 C28WNK 11682752 Ki = 3600 nM T86702 CKGR97 11692294 IC50 > 5000 nM T86702 C3U6ZR 11697504 Ki = 17000 nM T86702 C1MJ3P 11713694 IC50 = 756 nM T86702 C2BJ3X 11716217 Ki = 10000 nM T86702 C4ECU2 11720597 IC50 = 2157 nM T86702 CX91AZ 11723218 IC50 = 810 nM T86702 CBT48P 11731926 Ki = 10.7 nM T86702 CA43HK 11732287 Ki = 9.07 nM T86702 C7CED0 11733417 IC50 = 678 nM T86702 CI0KL2 11733573 IC50 = 5 nM T86702 C4HD9K 11751106 IC50 > 5000 nM T86702 CO8QT0 11753905 Ki = 54 nM T86702 C3N1WB 11754235 Ki = 3 nM T86702 C3P0TZ 11754739 Ki = 2900 nM T86702 CJ4G5D 11754907 IC50 = 18.7 nM T86702 CD6S0B 11757331 IC50 = 37280 nM T86702 CUC9R5 11758082 IC50 = 0.9 nM T86702 CZ5V9G 11758096 IC50 = 72 nM T86702 C3RW1X 11761191 Ki = 3 nM T86702 C63UAE 11761938 IC50 = 10000 nM T86702 C8K7IG 11779797 Ki = 3235.94 nM T86702 C04DFH 11783486 Ki = 13.2 nM T86702 CSY8N7 11792237 IC50 = 10000 nM T86702 CX59YU 11792994 IC50 = 7000 nM T86702 CKM6P2 11795228 IC50 = 71 nM T86702 CCSD72 11795621 IC50 = 6.918 nM T86702 C46KHU 11796490 IC50 = 7.3 nM T86702 C47OIA 11797154 IC50 = 10 nM T86702 CFQ09H 11797374 Ki = 71 nM T86702 CMX43N 11797375 Ki = 29 nM T86702 CJ4VL3 11797382 IC50 > 1000 nM T86702 CCD4W2 11797992 IC50 = 65 nM T86702 CHQR96 11798386 IC50 < 1 nM T86702 CGL39X 11798547 Ki = 520 nM T86702 CXFP23 11798966 IC50 = 18.2 nM T86702 CHS4I2 11800528 Ki = 24 nM T86702 CA82BI 11800904 Ki = 70 nM T86702 CCPL48 11811312 IC50 > 10000 nM T86702 CQ9HE2 11811551 IC50 = 4840 nM T86702 CSG07A 11811629 Ki > 650 nM T86702 CLW3F1 11812791 IC50 = 418 nM T86702 CH3SV6 11813493 IC50 = 316 nM T86702 CZ08ID 11814382 IC50 = 282 nM T86702 C8DY3Z 11817193 IC50 > 100000 nM T86702 C3VO5H 11824148 Ki = 9.8 nM T86702 CKEM29 11827006 IC50 = 26 nM T86702 C02BWA 11967143 Ki > 2000 nM T86702 CB80OT 12000718 IC50 = 8200 nM T86702 C43PJZ 12000720 IC50 = 15000 nM T86702 C0XKJ1 12671872 IC50 = 30000 nM T86702 C7C8FR 13875965 Ki = 52000 nM T86702 C1AJO7 13968141 IC50 > 300000 nM T86702 CA2H8V 14303060 IC50 = 20000 nM T86702 C1IZ7D 15296597 Ki = 86 nM T86702 CGH19T 15296844 IC50 > 300000 nM T86702 CK01NV 15379727 IC50 = 20 nM T86702 C63MFQ 15435266 IC50 = 16 nM T86702 CH80JI 15435267 Ki = 218.78 nM T86702 CZ0NL1 15484680 IC50 = 3400 nM T86702 COZM90 15485452 IC50 = 8 nM T86702 CEM2O0 15485453 IC50 = 3700 nM T86702 CT68FI 15487434 Ki = 1600 nM T86702 CJR3Z8 15487435 Ki = 370 nM T86702 C46XNB 15487436 Ki = 850 nM T86702 CV1HA9 15516783 IC50 = 150 nM T86702 C8B9QU 15546341 IC50 = 98 nM T86702 C5FA3L 15871222 IC50 = 0.7 nM T86702 CB3A4Z 15941413 Ki = 4100 nM T86702 CA40FE 15941550 Ki = 2200 nM T86702 CM3D1L 15941553 Ki = 12200 nM T86702 CQ0ZL7 15941677 Ki = 575 nM T86702 CV67UL 15986261 IC50 = 8700 nM T86702 C4VW5F 16058482 IC50 = 59 nM T86702 C4WX2I 16108938 IC50 > 1000 nM T86702 CD51GI 16108939 IC50 = 1200 nM T86702 C5YVB0 16108940 IC50 > 5000 nM T86702 CB4DU9 16108941 IC50 > 5000 nM T86702 CBW71J 16108942 IC50 > 5000 nM T86702 CG6R9L 16108943 IC50 > 3000 nM T86702 CN62KM 16108944 IC50 > 5000 nM T86702 C7YS5Q 16108947 IC50 > 5000 nM T86702 CLD2Y4 16108948 IC50 > 5000 nM T86702 CJR95O 16108949 IC50 > 1000 nM T86702 CRQ26L 16108950 IC50 > 5000 nM T86702 CH80AG 16108951 IC50 = 450 nM T86702 CWB0G9 16108952 IC50 > 1000 nM T86702 CQS0F5 16719301 IC50 = 1100 nM T86702 C75XDI 16730519 IC50 = 1800 nM T86702 C3S2TQ 17754305 IC50 = 5800 nM T86702 CQG89Z 17853548 IC50 = 58810 nM T86702 CK8FS7 18173159 IC50 = 62 nM T86702 CX10BM 18173179 IC50 = 69 nM T86702 CQO70Y 18173222 IC50 = 313 nM T86702 CXG1K2 18363133 IC50 > 10000 nM T86702 C37BNA 18363136 IC50 > 10000 nM T86702 C0KOW7 18363142 IC50 > 10000 nM T86702 CP04KS 18363146 IC50 > 10000 nM T86702 CLZD96 18363152 IC50 > 10000 nM T86702 CW3KB9 18363153 IC50 > 10000 nM T86702 CK30ZO 18363159 IC50 > 10000 nM T86702 CZU27R 18363164 IC50 > 10000 nM T86702 CC0UV8 18363169 IC50 > 10000 nM T86702 CR3CQ4 18363187 IC50 > 10000 nM T86702 CH5IU9 18363209 IC50 > 10000 nM T86702 CJGZ27 18363210 IC50 > 10000 nM T86702 CWI2A9 18363212 IC50 > 10000 nM T86702 C31LQZ 18363213 IC50 > 10000 nM T86702 CE60WD 18363216 IC50 > 10000 nM T86702 C3L6DU 18363223 IC50 > 10000 nM T86702 CD08XL 18379555 IC50 = 84 nM T86702 CXL6T9 18379569 IC50 = 51 nM T86702 C5LY6A 18379613 IC50 = 26 nM T86702 C0NLV5 18379626 IC50 = 205 nM T86702 CKY98M 18379668 IC50 = 6 nM T86702 CO21QH 18395616 IC50 = 550 nM T86702 C5B9WG 18533077 IC50 = 1200 nM T86702 CK5XU1 18666597 IC50 > 2 nM T86702 C2G6XM 18666600 IC50 = 210 nM T86702 C1GQ2O 18666601 IC50 = 1300 nM T86702 CYA3H7 18790040 IC50 > 10000 nM T86702 CBN28Y 18790155 Ki = 3300 nM T86702 CK8MP3 20620240 Ki = 8.7 nM T86702 CPC4G6 20620273 Ki = 37 nM T86702 C2E3CY 20620614 IC50 = 39 nM T86702 CA7FK0 20639531 IC50 = 860 nM T86702 CMX23W 20639537 IC50 = 490 nM T86702 C34XRP 20639540 IC50 = 550 nM T86702 C7AP8Z 20639546 IC50 = 500 nM T86702 CPK09X 20651316 IC50 = 0.7 nM T86702 CG1BD4 20689551 IC50 = 3100 nM T86702 C4I1OM 20735209 IC50 = 370 nM T86702 CT87YK 21699971 IC50 = 11000 nM T86702 CH4G5T 21699977 IC50 = 62 nM T86702 CQ1GI3 21699983 IC50 = 180000 nM T86702 CJZ58F 21699985 IC50 = 21000 nM T86702 CE72FU 21700004 IC50 = 120000 nM T86702 C5JC6W 21700038 IC50 = 36000 nM T86702 C3QAP8 21700080 IC50 = 17000 nM T86702 CG0RI5 21700124 IC50 = 4000 nM T86702 CXME27 21700151 IC50 = 37000 nM T86702 CFK4Y7 21700160 IC50 = 35000 nM T86702 CIJ93L 21700163 IC50 = 37000 nM T86702 CB1QH3 21700191 IC50 = 300000 nM T86702 CUVE24 21700204 IC50 = 130000 nM T86702 C36WFA 22096205 IC50 > 100000 nM T86702 CZT05X 22484417 Ki = 900 nM T86702 CZT64B 22484431 Ki = 31 nM T86702 CAM10T 22485252 IC50 = 55.3 nM T86702 CAY3N6 22485292 IC50 = 22.5 nM T86702 C3YL5X 22485311 IC50 = 32.6 nM T86702 CWA03L 22485327 IC50 = 20.6 nM T86702 C5JZF1 22485344 IC50 = 35 nM T86702 CI7MY5 22485346 IC50 = 50 nM T86702 CI1YL7 22485347 IC50 = 20 nM T86702 C25OBD 22485356 IC50 = 18.1 nM T86702 CL64TJ 22485368 IC50 = 36.9 nM T86702 CT4GF9 22485381 IC50 = 550 nM T86702 C27NDB 22485386 IC50 = 64.7 nM T86702 C3MG9P 22485396 IC50 = 35 nM T86702 CZY10U 22485408 IC50 = 40 nM T86702 C89AGT 22485413 IC50 = 18.1 nM T86702 C03NLM 22485417 IC50 = 7 nM T86702 C8GHU9 22485432 IC50 = 21.5 nM T86702 CWPM36 22642543 IC50 = 10 nM T86702 C5EQ7I 22642544 IC50 = 80 nM T86702 CD71UM 22642553 IC50 = 20 nM T86702 CRL2G4 22642563 IC50 = 30 nM T86702 C2Q4XK 22707806 IC50 = 18.1 nM T86702 CA59OL 22856307 Ki = 1300 nM T86702 CK6IM2 22907131 Ki = 134 nM T86702 CVF9M4 22922043 IC50 = 38150 nM T86702 CX2JO7 22950015 IC50 = 7.244 nM T86702 CIYA45 22985930 IC50 = 21.5 nM T86702 CF75MS 23017979 IC50 = 5500 nM T86702 CQJ3S4 23018008 IC50 = 2000 nM T86702 CM5H2P 23061661 IC50 > 10000 nM T86702 C97LAR 23061665 IC50 > 10000 nM T86702 C9GKH3 23523881 IC50 = 20 nM T86702 CU8O7L 23523890 IC50 = 30 nM T86702 CSXG85 23523891 IC50 = 20 nM T86702 CV85UI 23523893 IC50 = 400 nM T86702 CXZ20T 23523894 IC50 = 300 nM T86702 CPLS94 23523896 IC50 = 10000 nM T86702 CM0K4X 23523897 IC50 = 100 nM T86702 CBI65T 23523899 IC50 = 10000 nM T86702 CP6ZF2 23523900 IC50 = 100 nM T86702 CGWL84 23523905 IC50 = 400 nM T86702 CY7RC8 23523909 IC50 = 20 nM T86702 CV06HF 23523910 IC50 = 6000 nM T86702 CU8BN9 23523911 IC50 = 500 nM T86702 C5GR7Y 23523914 IC50 = 700 nM T86702 C4R2DA 23645953 Ki > 300000 nM T86702 CWN3I4 23645959 Ki > 300000 nM T86702 C6AW7U 23692637 IC50 > 100000 nM T86702 CQCJ17 24768595 IC50 = 39 nM T86702 C5M3YW 24799779 Ki = 58000 nM T86702 C9RW0A 24806176 IC50 = 137 nM T86702 C18FRG 24807817 IC50 = 25000 nM T86702 CW3X0F 24852010 IC50 = 79.1 nM T86702 C6YPS8 24852048 IC50 = 56.5 nM T86702 C4UEM5 24871537 Ki > 50000 nM T86702 CP2L5B 24871655 Ki > 50000 nM T86702 C9K5WP 24879338 IC50 = 610 nM T86702 CFL04M 24881245 IC50 > 300000 nM T86702 CLIC14 24881246 IC50 > 300000 nM T86702 C4FI5C 24901479 IC50 = 38 nM T86702 C4SP3O 24936157 IC50 = 105 nM T86702 CBUA83 24936183 IC50 = 203 nM T86702 CQ2K9H 24936215 IC50 > 5000 nM T86702 C0EA5F 24936382 IC50 = 0.038 nM T86702 CNCA57 25004194 Ki = 4500 nM T86702 CAQ9Z1 25022681 Ki > 4501 nM T86702 CVR52U 25066764 IC50 = 351 nM T86702 CD2KA4 25102047 IC50 = 450 nM T86702 CRW96X 25102048 IC50 = 71 nM T86702 CQ3O9P 25102050 IC50 = 47 nM T86702 CSHA26 25102051 IC50 = 120 nM T86702 C7ADO2 25102197 IC50 = 36 nM T86702 CA5DJ4 25138228 Ki < 14000 nM T86702 C6N7EQ 25138258 Ki = 2970 nM T86702 C7AD1J 25138259 Ki = 852 nM T86702 CJ9TQ2 25138260 Ki = 3690 nM T86702 CUT8I7 25138261 Ki = 3060 nM T86702 CBD9X6 25138262 Ki = 1123 nM T86702 C8LX1S 25138263 Ki = 627 nM T86702 C3OV1L 25138264 Ki = 2719 nM T86702 C92WVM 25138265 Ki = 766 nM T86702 CMCS41 25138266 Ki > 4501 nM T86702 C1FJV5 25138267 Ki > 4501 nM T86702 C9N6WT 25138268 Ki > 4501 nM T86702 CF4QI1 25138269 Ki > 4501 nM T86702 C6P5UL 25138270 Ki = 3306 nM T86702 CQE0L7 25138271 Ki = 3305 nM T86702 C59XWU 25138272 Ki > 4501 nM T86702 C1TNQ3 25141117 Ki = 415 nM T86702 CR35QP 25144971 IC50 < 100 nM T86702 C0Y5BC 25145683 IC50 > 2500 nM T86702 CEP9Q2 25180867 IC50 = 6.7 nM T86702 C6EWF1 25183622 Ki > 10000 nM T86702 CAH7T2 25183623 Ki > 10000 nM T86702 CXG2S6 25183625 Ki > 10000 nM T86702 CHR2P1 25183768 Ki > 25000 nM T86702 C1HZ9E 40424573 Ki = 120000 nM T86702 C8KM4E 43366432 IC50 > 10000 nM T86702 CPO1Z3 44123600 IC50 = 18 nM T86702 CH1IR0 44144307 IC50 = 25550 nM T86702 CT80ED 44219901 IC50 = 1800 nM T86702 C94JVY 44219902 IC50 = 710 nM T86702 C7J6GH 44219903 IC50 = 1200 nM T86702 C9J7WL 44219904 IC50 = 4300 nM T86702 CRQ71E 44219905 IC50 = 9100 nM T86702 C4Z0ID 44219906 IC50 = 4300 nM T86702 CRNA25 44220092 IC50 = 1200 nM T86702 C9T5ZF 44220093 IC50 = 180 nM T86702 CV38TE 44222825 IC50 = 1600 nM T86702 CJI73R 44222826 IC50 = 1300 nM T86702 CGQ30N 44222827 IC50 = 1800 nM T86702 CCI64J 44224245 IC50 = 300 nM T86702 CLRT69 44247751 IC50 = 21 nM T86702 CAR34Y 44263877 IC50 = 404 nM T86702 CEV08N 44263913 IC50 = 14 nM T86702 C5ZI0X 44263926 IC50 = 3.3 nM T86702 CO3C1E 44263994 IC50 = 39.2 nM T86702 C9XJ7U 44264020 IC50 = 180 nM T86702 C6L0MJ 44264021 IC50 = 6.5 nM T86702 CJ1WE7 44264036 IC50 = 3.5 nM T86702 C50QFR 44264375 IC50 = 5.3 nM T86702 C4C7DY 44265493 Ki = 15 nM T86702 CXSD62 44265506 Ki = 68 nM T86702 CC5WJ2 44265518 Ki = 38 nM T86702 COY0U7 44265581 Ki = 82 nM T86702 COU3Y8 44266817 IC50 = 3700 nM T86702 CUA5E0 44266818 IC50 = 5100 nM T86702 CG23BI 44266830 IC50 = 4270 nM T86702 C3HP1F 44270658 IC50 = 4100 nM T86702 CQAY10 44270663 IC50 = 28 nM T86702 CRX9Z2 44270670 IC50 = 140 nM T86702 C8S2FJ 44270678 IC50 = 130 nM T86702 C2BUH0 44270679 IC50 = 39 nM T86702 C4C3RN 44270683 IC50 = 290 nM T86702 C4OJK9 44270703 IC50 = 43 nM T86702 C8MUJ3 44270704 IC50 = 110 nM T86702 C7CVT3 44270713 IC50 = 22 nM T86702 CQTE41 44270720 IC50 = 210 nM T86702 CCDW47 44270721 IC50 = 860 nM T86702 C96OIC 44270729 IC50 = 140 nM T86702 CRP24X 44270733 IC50 = 13 nM T86702 C0K3RP 44270736 IC50 = 88 nM T86702 CLMO84 44270737 IC50 = 160 nM T86702 CKL2C3 44270739 IC50 = 26 nM T86702 C47OXE 44270748 IC50 = 120 nM T86702 C4B0LP 44270775 IC50 = 5100 nM T86702 CYZX59 44270776 IC50 = 1500 nM T86702 C9CXP4 44270786 IC50 = 120 nM T86702 C1WTN7 44270802 IC50 = 88 nM T86702 C6UQ8N 44270804 IC50 > 20 nM T86702 CVG61X 44270805 IC50 = 4600 nM T86702 CNU41R 44270901 IC50 = 36 nM T86702 CDX36Y 44270985 IC50 = 39 nM T86702 CFR81A 44271005 IC50 = 430 nM T86702 CG7X5F 44272675 IC50 = 4.4 nM T86702 CEHR24 44272853 IC50 = 61 nM T86702 CA6OU2 44273333 Ki = 280 nM T86702 C9S6GJ 44273334 Ki = 710 nM T86702 CU1D5I 44273335 Ki = 560 nM T86702 C04LMN 44273336 Ki = 340 nM T86702 CU2L9K 44273556 Ki = 15 nM T86702 COV24P 44273558 Ki = 1400 nM T86702 C2UBY7 44273577 Ki = 1300 nM T86702 CV6T9M 44273670 Ki = 280 nM T86702 C1FAV6 44273674 Ki = 370 nM T86702 C2FH5M 44273675 Ki = 4600 nM T86702 C13WVU 44273676 Ki = 600 nM T86702 COHD62 44273677 Ki = 210 nM T86702 CQ2N5J 44273682 Ki = 410 nM T86702 C2RA8T 44273710 Ki = 20 nM T86702 C4SHN1 44273711 Ki = 6.1 nM T86702 CESY58 44273712 Ki = 24 nM T86702 CO0E8C 44273725 Ki = 2400 nM T86702 CO79TR 44273726 Ki = 330 nM T86702 CA7NY1 44273727 Ki = 940 nM T86702 CYL2B4 44273802 Ki = 42 nM T86702 C8CB4A 44275752 IC50 = 1200 nM T86702 CVI56W 44275768 IC50 = 2700 nM T86702 C2MWR0 44275913 Ki = 62 nM T86702 CKV1E7 44275972 Ki = 1.4 nM T86702 C6YT3K 44280285 Ki = 6575 nM T86702 C8XUJ3 44280321 Ki = 25000 nM T86702 CC2O3U 44280323 Ki = 806 nM T86702 CM2TZ4 44280335 Ki > 800 nM T86702 CA1V6Y 44280345 Ki = 15 nM T86702 C8KZ2F 44281541 IC50 = 170 nM T86702 CRK8H6 44281557 IC50 = 420 nM T86702 CTJ7Q2 44281563 IC50 = 480 nM T86702 COU71D 44281564 IC50 = 160 nM T86702 CJ2PG9 44281705 IC50 = 15 nM T86702 CC2QR7 44281720 Ki = 267 nM T86702 C1M3JR 44281777 IC50 = 95 nM T86702 CL18QW 44281786 IC50 = 91 nM T86702 C3ES4Z 44281796 IC50 = 50 nM T86702 C60HIN 44281797 IC50 = 170 nM T86702 C8U5GR 44281941 IC50 = 2600 nM T86702 CN23FC 44282968 IC50 = 2500 nM T86702 C2TV5I 44282969 IC50 = 350 nM T86702 CG3LF0 44282970 IC50 > 2000 nM T86702 C4LKS7 44285342 Ki = 119000 nM T86702 CCL4F1 44285343 IC50 = 173000 nM T86702 COY3I9 44285516 Ki = 85000 nM T86702 C6JLI2 44285620 Ki = 420 nM T86702 CBZE45 44285686 IC50 = 97000 nM T86702 CXT37W 44286406 IC50 > 100000 nM T86702 C7CU3J 44286466 IC50 = 45000 nM T86702 CZ2AL1 44286483 IC50 = 80000 nM T86702 C3UB9V 44286654 Ki = 58.05 nM T86702 CB07MX 44286663 Ki = 11.5 nM T86702 C3KXY9 44286674 Ki = 0.43 nM T86702 C96NMF 44287796 IC50 = 320 nM T86702 CQ5IG7 44287805 IC50 = 68 nM T86702 CHOV34 44287806 IC50 = 320 nM T86702 CYAG29 44287899 IC50 = 8 nM T86702 CX5QB3 44287917 IC50 = 20 nM T86702 CCM31I 44288043 IC50 = 30 nM T86702 C1YT7H 44288071 IC50 = 29 nM T86702 CF2DZ9 44288091 IC50 = 5900 nM T86702 CMY2N4 44288092 IC50 = 112 nM T86702 CCS20R 44288093 IC50 = 5 nM T86702 CJ1HT6 44288855 IC50 > 10000 nM T86702 CT38HI 44289140 IC50 > 10000 nM T86702 CAH30U 44289181 IC50 > 10000 nM T86702 CH1TS5 44289182 IC50 > 10000 nM T86702 CMZ2O6 44289200 IC50 > 10000 nM T86702 CBLC60 44289352 Ki = 734 nM T86702 CZO75J 44289369 Ki = 60 nM T86702 CRT7O2 44289382 Ki = 86 nM T86702 C7WUJ2 44289459 IC50 > 10000 nM T86702 CJ73FW 44289479 IC50 > 10000 nM T86702 CWMI67 44289482 IC50 > 10000 nM T86702 C1L4ZU 44289489 IC50 > 10000 nM T86702 C19EJM 44289515 IC50 > 10000 nM T86702 C6TI3X 44289520 Ki > 10000 nM T86702 CA52ED 44289521 Ki > 10000 nM T86702 C30KSP 44289579 Ki = 1430 nM T86702 CHC08W 44289601 Ki = 590 nM T86702 CZ4EI7 44289602 Ki = 300 nM T86702 CEML82 44289603 Ki = 4420 nM T86702 CM26JT 44289604 Ki = 676 nM T86702 CLY4K5 44289640 Ki = 184 nM T86702 C7GY8M 44289643 Ki > 10000 nM T86702 CV9B2F 44289867 Ki > 10000 nM T86702 CJ7VW3 44291166 IC50 = 0.7 nM T86702 C75IEN 44291420 IC50 = 20 nM T86702 C51TQK 44291531 IC50 = 90 nM T86702 CF21CS 44291532 IC50 = 37 nM T86702 CU75TB 44291559 IC50 = 45 nM T86702 C06JAO 44291626 IC50 = 29 nM T86702 C4LI6F 44293416 Ki = 1.93 nM T86702 C5XS0I 44294322 Ki = 14088 nM T86702 C1Q9VY 44294552 Ki = 552 nM T86702 CO51MC 44294736 IC50 > 200000 nM T86702 C3A0JQ 44294777 Ki = 77 nM T86702 CO29ZW 44294804 IC50 > 200000 nM T86702 CMF09R 44294805 Ki = 550 nM T86702 CM7Q5H 44294856 Ki = 42 nM T86702 CICM29 44294857 IC50 = 81 nM T86702 CTR80J 44294877 IC50 = 55000 nM T86702 C4JI5K 44299989 IC50 = 100 nM T86702 C5RSX9 44300181 IC50 = 38000 nM T86702 COW30X 44300184 IC50 = 10000 nM T86702 CI13FM 44300231 IC50 = 400 nM T86702 CKN3P7 44302022 IC50 = 2000 nM T86702 C2Y0PK 44302023 IC50 = 1250 nM T86702 C5S3UO 44302024 IC50 = 230 nM T86702 C8ERW6 44302042 IC50 = 410 nM T86702 C6JXH0 44302043 IC50 = 7000 nM T86702 CI56DL 44302044 IC50 = 4000 nM T86702 CWB83G 44302076 IC50 = 320 nM T86702 CY1J9U 44302096 IC50 = 520 nM T86702 CW94ZQ 44302164 IC50 = 4700 nM T86702 C2FSR6 44302165 IC50 = 18 nM T86702 CQ54PZ 44302166 IC50 = 50 nM T86702 C9U3XT 44302167 IC50 = 90 nM T86702 C5X1WY 44302183 IC50 = 783 nM T86702 C7G3BN 44302200 IC50 = 2320 nM T86702 CMB4Q8 44302221 IC50 = 5000 nM T86702 C70QWV 44302327 IC50 = 30000 nM T86702 CZP20C 44302339 IC50 = 600 nM T86702 CO73BW 44302357 IC50 = 630 nM T86702 C6R0VK 44302358 IC50 = 1000 nM T86702 CXUZ19 44302359 IC50 = 40 nM T86702 CNL4E2 44302361 IC50 = 300 nM T86702 CCW65Y 44302378 IC50 = 1001 nM T86702 CDK9W1 44302383 IC50 = 80 nM T86702 CYG80V 44302385 IC50 = 500 nM T86702 C7ZBR4 44302396 IC50 = 450 nM T86702 C8S5WT 44302397 IC50 = 40 nM T86702 CPC25G 44302409 IC50 = 1610 nM T86702 C4QL0I 44302411 IC50 = 30 nM T86702 C4NDA2 44302416 IC50 = 1340 nM T86702 C24ZWF 44302429 IC50 = 560 nM T86702 C4I6WO 44302430 IC50 = 70 nM T86702 CYL71W 44302432 IC50 = 60 nM T86702 C5H6OV 44302627 IC50 = 2150 nM T86702 C6QR7C 44302634 IC50 = 860 nM T86702 CG8KJ0 44302661 IC50 = 250 nM T86702 CUZS20 44302663 IC50 = 20000 nM T86702 CX1M3Q 44302666 IC50 = 210 nM T86702 C36CQP 44302952 IC50 = 500 nM T86702 C0IJ9D 44304112 Ki = 7.29 nM T86702 C7ME6Z 44305408 IC50 = 58 nM T86702 CD9W5Q 44305414 IC50 = 215 nM T86702 CY18UG 44305656 IC50 = 250 nM T86702 C4QIF8 44305668 IC50 = 1420 nM T86702 CA0GN1 44305669 IC50 = 518 nM T86702 CNF86G 44305670 IC50 = 21 nM T86702 CXF6Y3 44305706 IC50 = 11700 nM T86702 CCHK59 44305722 IC50 = 824 nM T86702 C6EZU9 44305732 IC50 = 2900 nM T86702 C4ZI6D 44305743 IC50 = 104 nM T86702 CI82ZH 44305746 IC50 = 30 nM T86702 CLK31H 44305747 IC50 = 108 nM T86702 COI82F 44305750 IC50 = 94 nM T86702 CLH14M 44305978 IC50 = 12 nM T86702 CZ49UN 44305988 IC50 = 6.1 nM T86702 CO2SK0 44306005 Ki = 13 nM T86702 C6I8JA 44306058 IC50 = 6.9 nM T86702 CB5EY3 44306200 IC50 = 12 nM T86702 C0YOH1 44306202 IC50 = 4.2 nM T86702 CMA39E 44306203 IC50 = 2.6 nM T86702 CL58OS 44306208 IC50 = 2100 nM T86702 CAY2S4 44306209 IC50 = 75 nM T86702 C27NJX 44306277 IC50 = 1.8 nM T86702 C6O1AN 44306279 IC50 = 9.1 nM T86702 C5QUK2 44308295 Ki = 354 nM T86702 C2E4IT 44308297 Ki = 120 nM T86702 C0K4UQ 44308298 Ki = 93 nM T86702 CCRW50 44308304 Ki = 80 nM T86702 CZF5S2 44308327 Ki = 153 nM T86702 COE56H 44308377 Ki = 2323 nM T86702 C7OT6S 44308488 Ki = 406 nM T86702 CI2Z0H 44308525 Ki = 135 nM T86702 CU0J5A 44308623 Ki = 38 nM T86702 CSEB94 44308624 Ki = 45 nM T86702 CST39W 44308640 Ki = 437 nM T86702 CKEU31 44309629 IC50 = 19000 nM T86702 CJ9OE7 44313735 IC50 = 47 nM T86702 C5HAY4 44313736 IC50 = 9.1 nM T86702 CX4BM9 44313996 IC50 = 2175 nM T86702 C5ZTU6 44314442 Ki = 321 nM T86702 C2JUX9 44314443 Ki = 353 nM T86702 CC95EZ 44314744 Ki = 25.3 nM T86702 CY63DG 44314754 Ki = 1.73 nM T86702 C8ZD7F 44314755 Ki = 834 nM T86702 COF0B1 44314762 Ki = 8.24 nM T86702 C59CBZ 44314763 Ki = 8.3 nM T86702 C9L1NY 44314788 Ki = 2.75 nM T86702 CM04TG 44314789 Ki = 6.35 nM T86702 C7LCN0 44314824 Ki = 358 nM T86702 CNM6W8 44314841 Ki = 0.8 nM T86702 C9K8JZ 44314900 Ki = 177 nM T86702 CXRE70 44314901 Ki = 4.16 nM T86702 CK3H1Y 44314929 Ki = 77 nM T86702 CS5A6Z 44314930 Ki = 13.5 nM T86702 CNB72W 44314931 Ki = 22.2 nM T86702 CBXI30 44314932 Ki = 2.61 nM T86702 CCF80X 44314958 Ki = 8400 nM T86702 C3N8RQ 44314969 Ki = 1110 nM T86702 C9SRT4 44314970 Ki = 358 nM T86702 C61DST 44314974 Ki = 2.39 nM T86702 CE2J4M 44314975 Ki = 6.26 nM T86702 CQE0D3 44314976 Ki = 81.5 nM T86702 CI2V1Y 44314995 Ki = 3120 nM T86702 C48NVD 44314999 Ki = 0.96 nM T86702 CB7F0J 44315000 Ki = 90.3 nM T86702 CDZ5O3 44315029 Ki = 2200 nM T86702 C6HW5G 44315084 Ki = 2.98 nM T86702 CV6KW1 44315085 Ki = 1.38 nM T86702 CH48TD 44315155 IC50 = 2700 nM T86702 CAUQ47 44315167 Ki = 1470 nM T86702 COA01P 44315179 Ki = 19100 nM T86702 CQ1R9E 44315204 Ki = 1060 nM T86702 CL32FZ 44315221 Ki = 4100 nM T86702 CDN4Y5 44315222 Ki = 29400 nM T86702 C62FXJ 44315244 IC50 = 900 nM T86702 CP9M6W 44315277 Ki = 5.44 nM T86702 C3SZO4 44315279 Ki = 701 nM T86702 CSG05N 44315321 Ki = 5.87 nM T86702 COD08C 44315324 Ki = 952 nM T86702 C50IQE 44315333 IC50 = 800 nM T86702 C37JMW 44315348 Ki = 952 nM T86702 C8Y7JG 44317981 Ki = 4677.35 nM T86702 C89IQW 44318090 IC50 = 86.1 nM T86702 C6FG7Y 44322562 IC50 = 800 nM T86702 CK0T6M 44322564 IC50 = 900 nM T86702 C0QJE9 44322722 IC50 = 900 nM T86702 C90EGJ 44322757 IC50 = 900 nM T86702 CO0S9J 44325072 Ki = 1.8 nM T86702 C4R9LM 44325085 Ki = 2.6 nM T86702 CL8MD0 44325156 Ki = 42 nM T86702 CV3S9G 44325157 Ki = 85 nM T86702 C9MD1A 44325159 Ki = 490 nM T86702 C6R4NI 44325225 Ki = 44 nM T86702 C3M2XY 44325277 Ki = 1.7 nM T86702 CA4FQ5 44325443 Ki = 50 nM T86702 C20UGO 44325517 Ki > 10000 nM T86702 CHMC02 44325564 Ki = 20000 nM T86702 C8P6UA 44325625 Ki = 2.61 nM T86702 CBY75J 44325686 Ki > 10000 nM T86702 C6A1JX 44325696 Ki = 22.2 nM T86702 CJU3R8 44325730 Ki = 0.96 nM T86702 CBV73K 44325744 Ki = 2.39 nM T86702 C06ZAH 44325745 Ki = 6.26 nM T86702 C70UFH 44325749 Ki = 1.38 nM T86702 C8EWP2 44325750 Ki = 5.87 nM T86702 C2QL0B 44325810 Ki = 6.35 nM T86702 CP1NU9 44325834 Ki = 8.15 nM T86702 C7VRX2 44325907 Ki = 0.8 nM T86702 C7V5EF 44326167 IC50 = 970 nM T86702 C93HSL 44326184 IC50 = 1400 nM T86702 CY3I9B 44326185 IC50 = 45 nM T86702 C23OQF 44326225 IC50 = 270 nM T86702 CY3GH5 44326232 IC50 = 4280 nM T86702 C6E9IV 44326443 IC50 = 2600 nM T86702 C85QTP 44328155 IC50 = 90000 nM T86702 CZQ6N7 44328189 IC50 = 1000 nM T86702 CBD0Z2 44329014 IC50 = 2340 nM T86702 CMLA39 44329018 IC50 = 179 nM T86702 C84MVU 44329019 IC50 = 665 nM T86702 C90CHA 44329405 IC50 = 7000 nM T86702 CI3Z4K 44329623 IC50 = 60 nM T86702 C6OL8M 44329636 IC50 = 3981.07 nM T86702 CA65RO 44329672 IC50 = 1995.26 nM T86702 CK9HO7 44329673 IC50 = 5000 nM T86702 C07GRS 44329693 IC50 = 60 nM T86702 CBH16R 44329694 IC50 = 398.11 nM T86702 CG3E7A 44329712 IC50 = 7 nM T86702 C9SN6I 44329713 IC50 = 6000 nM T86702 CZ2FW6 44329725 IC50 = 1995.26 nM T86702 CDKI48 44329741 IC50 = 800 nM T86702 CK3M2H 44329742 IC50 = 10000 nM T86702 C39RDS 44329886 IC50 = 50 nM T86702 C3YAF6 44329898 IC50 = 1500 nM T86702 C63RHP 44329909 IC50 = 100 nM T86702 CVQA75 44329910 IC50 = 794.33 nM T86702 C84SLI 44329926 IC50 = 30 nM T86702 CJS6B1 44329927 IC50 = 300 nM T86702 C9R1ZE 44330132 IC50 = 10000 nM T86702 CLU8I7 44330135 IC50 = 280 nM T86702 C1IE0S 44330147 IC50 = 10000 nM T86702 CPG7N2 44330149 IC50 = 1300 nM T86702 CYP6S4 44330152 IC50 = 1200 nM T86702 CMGA28 44330163 IC50 = 6300 nM T86702 CG2Q8W 44332306 IC50 = 71 nM T86702 C5RMC9 44333946 IC50 = 300 nM T86702 CZ8P6F 44333947 IC50 = 9670 nM T86702 CCF9D5 44333961 IC50 = 20400 nM T86702 CLVH73 44333962 IC50 = 2700 nM T86702 C5NG0R 44334948 IC50 = 20 nM T86702 CFP3X8 44334949 IC50 = 45 nM T86702 CV5RF0 44334963 IC50 = 293 nM T86702 C4AOZ7 44334981 IC50 = 136 nM T86702 CXW59C 44334982 IC50 = 16.7 nM T86702 CCH1W8 44334983 IC50 = 3 nM T86702 CQ0UI1 44335017 IC50 = 10.1 nM T86702 CX58SB 44335240 IC50 = 6.7 nM T86702 CA96JG 44335285 IC50 = 6.5 nM T86702 CM3F2G 44337397 IC50 = 3000 nM T86702 C9L3HU 44337570 IC50 = 3000 nM T86702 CI5X0G 44339523 IC50 = 7.2 nM T86702 CB9K8T 44339536 IC50 = 8.9 nM T86702 C2R3XN 44339554 IC50 = 3.2 nM T86702 C2CRY1 44339556 IC50 = 10 nM T86702 CTBU53 44339564 IC50 = 36 nM T86702 C58OSK 44339567 IC50 = 1.8 nM T86702 CX2KJ3 44339574 IC50 = 54 nM T86702 CEK3G0 44339588 IC50 = 9.8 nM T86702 C7ZR6H 44339589 IC50 = 360 nM T86702 C0WP9C 44339590 IC50 = 6.6 nM T86702 C5C2LI 44339654 IC50 = 5.6 nM T86702 CH3I5B 44339870 Ki = 670 nM T86702 CM6VJ2 44339884 Ki = 170 nM T86702 CMVE19 44339885 Ki = 540 nM T86702 CLD2P9 44339900 Ki = 440 nM T86702 C5R6KD 44339905 Ki = 470 nM T86702 C3B5XK 44339917 Ki = 24 nM T86702 C2D6VN 44339918 Ki = 13 nM T86702 CRQJ09 44339936 Ki = 520 nM T86702 CNED21 44340075 Ki = 410 nM T86702 C07CVA 44340076 IC50 = 2800 nM T86702 C4JLG8 44340091 Ki = 62 nM T86702 CLKT58 44340092 Ki = 50 nM T86702 C4KLU8 44340093 Ki = 70 nM T86702 CXW34P 44340094 Ki = 17 nM T86702 CZ45CH 44340125 IC50 = 260 nM T86702 CZ98KU 44340156 Ki = 130 nM T86702 C7E5FI 44340159 Ki = 54 nM T86702 CGV94P 44340160 Ki = 5.5 nM T86702 C3IS1O 44340161 Ki = 30 nM T86702 CPK5W0 44340172 Ki = 5.7 nM T86702 C4SC6L 44340175 IC50 > 200000 nM T86702 CVJM53 44340176 IC50 = 430 nM T86702 CDR5V6 44340199 Ki = 63 nM T86702 C7PAI6 44340200 Ki = 56 nM T86702 CJ4Z9W 44340207 Ki = 1500 nM T86702 CZ31VY 44340208 Ki = 2.3 nM T86702 CVG1R5 44340217 Ki = 16 nM T86702 C39EMX 44340229 Ki = 3700 nM T86702 C4B9QZ 44340327 Ki = 1.4 nM T86702 C2XY8H 44340328 Ki = 2.5 nM T86702 CUM9J0 44340329 Ki = 26 nM T86702 CAT48Z 44340657 Ki = 33 nM T86702 CJBC96 44340662 Ki = 120 nM T86702 CJ83VB 44340663 Ki = 190 nM T86702 C3CYZ8 44340673 Ki = 350 nM T86702 CRI8Q4 44340696 Ki = 320 nM T86702 CF1QZ3 44340718 Ki = 28 nM T86702 C09ILT 44340727 Ki = 32 nM T86702 CSE9X6 44340728 Ki = 120 nM T86702 C6AS8J 44340740 Ki = 140 nM T86702 CAC07H 44340742 Ki = 130 nM T86702 CPVL28 44340743 Ki = 120 nM T86702 CH8BO5 44340744 Ki = 180 nM T86702 CQ4RT5 44340809 Ki = 110 nM T86702 CL0U9T 44340810 Ki = 10 nM T86702 CE4J9N 44340811 Ki = 270 nM T86702 CV6W7Z 44340812 Ki = 270 nM T86702 C3WZM0 44340828 Ki = 530 nM T86702 CW53EF 44340868 Ki = 47 nM T86702 C6ZDV3 44340869 Ki = 20 nM T86702 CR1ID4 44340923 Ki = 12 nM T86702 C2XP4N 44342352 Ki = 18 nM T86702 CURT86 44342353 Ki = 30 nM T86702 C2SZB1 44342614 IC50 = 200 nM T86702 CD1EL8 44344025 IC50 = 340 nM T86702 C8G7WL 44344564 Ki = 1700 nM T86702 CD43AB 44344565 Ki = 2700 nM T86702 CTQ6P4 44344631 IC50 = 23 nM T86702 CBH9I5 44344658 IC50 = 2.1 nM T86702 CC29QO 44344739 Ki = 3500 nM T86702 CWA42F 44344746 Ki = 39 nM T86702 CQPN17 44344749 Ki = 11 nM T86702 CL41FG 44344753 Ki = 40000 nM T86702 CF2IP7 44349785 IC50 > 20000 nM T86702 C4NUE8 44349786 IC50 = 18000 nM T86702 CCF94Z 44349787 IC50 = 9.4 nM T86702 CXY8T0 44349796 IC50 = 14000 nM T86702 C8P5UH 44349797 IC50 > 20000 nM T86702 C4SDB9 44349809 IC50 = 1100 nM T86702 C4PZL1 44349812 IC50 > 20000 nM T86702 C97GQR 44349822 IC50 > 20000 nM T86702 C2ZA6M 44349824 IC50 > 20000 nM T86702 CZ3LS0 44349842 IC50 = 550 nM T86702 C8X5LF 44349860 IC50 = 1900 nM T86702 CS95MA 44349861 IC50 = 510 nM T86702 C1L2GF 44350073 IC50 = 216 nM T86702 CQ5RN6 44350101 IC50 = 21 nM T86702 CE2X3Q 44350116 IC50 > 100 nM T86702 CD96OP 44356667 IC50 ~ 100000 nM T86702 C83BTI 44356670 Ki = 1600 nM T86702 CH4V6J 44356671 Ki = 640 nM T86702 CO5XG6 44356688 IC50 = 27300 nM T86702 CZQF75 44356702 IC50 = 6500 nM T86702 C1A4NY 44356703 IC50 = 10800 nM T86702 C4NM2V 44356737 Ki = 230 nM T86702 CE81GS 44356767 IC50 = 22000 nM T86702 C0BRH3 44356774 IC50 = 27000 nM T86702 C4G3KR 44356775 IC50 = 47000 nM T86702 C9DIQ5 44356789 IC50 > 100000 nM T86702 CO3RI0 44356790 IC50 = 28000 nM T86702 C8XA0M 44356791 IC50 = 12000 nM T86702 CCY5U3 44356804 Ki = 6.5 nM T86702 C25ZQU 44356805 IC50 > 100000 nM T86702 C1YAR5 44356962 Ki = 590 nM T86702 C2Y4KQ 44356963 Ki > 10000 nM T86702 CJH1C3 44356964 Ki = 110 nM T86702 CEI0X5 44357004 IC50 = 42000 nM T86702 C1LE9J 44359497 IC50 = 6000 nM T86702 CHE08D 44359498 IC50 = 10000 nM T86702 C4Z5RV 44359507 IC50 = 20 nM T86702 C2HZ6K 44359536 IC50 = 700 nM T86702 C1J4KA 44359537 IC50 = 3000 nM T86702 CV4ZM1 44359563 IC50 = 50 nM T86702 CP1CD9 44359641 IC50 = 20 nM T86702 CI5FY8 44359659 IC50 = 10 nM T86702 CJB74Y 44359661 IC50 = 30 nM T86702 CC9LH6 44359662 IC50 = 10000 nM T86702 CHW43J 44359663 IC50 = 2000 nM T86702 C17QMW 44359665 IC50 = 10000 nM T86702 CKD2L0 44359666 IC50 = 500 nM T86702 CJ2QU8 44359668 IC50 = 1000 nM T86702 CKM4W6 44359670 IC50 = 10000 nM T86702 CC7UB0 44359671 IC50 = 200 nM T86702 CJ91ZQ 44359676 IC50 = 10000 nM T86702 CY4CA6 44359677 IC50 = 40 nM T86702 C92OKL 44359678 IC50 = 100 nM T86702 CHWK87 44359686 IC50 = 10000 nM T86702 CEDO94 44359692 IC50 = 30 nM T86702 CC96HP 44359693 IC50 = 300 nM T86702 CHZK92 44359695 IC50 = 10000 nM T86702 C6XBP4 44359701 IC50 = 900 nM T86702 C2C7LJ 44359712 IC50 = 20 nM T86702 CVA09S 44359714 IC50 = 10000 nM T86702 CNX27J 44359717 IC50 = 400 nM T86702 CLG0O4 44359719 IC50 = 1000 nM T86702 CZL92R 44359720 IC50 = 1000 nM T86702 C3T0BS 44359739 IC50 = 2000 nM T86702 CCN30T 44359740 IC50 = 600 nM T86702 C3NIL4 44359744 IC50 = 600 nM T86702 CR7E8B 44359745 IC50 = 200 nM T86702 CP02BN 44359746 IC50 = 700 nM T86702 CX65KF 44359747 IC50 = 20 nM T86702 C8PKH7 44359748 IC50 = 600 nM T86702 CJ41AC 44359758 IC50 = 10000 nM T86702 CNSL71 44359759 IC50 = 500 nM T86702 CZ4E9Q 44359760 IC50 = 500 nM T86702 C7NTP1 44359790 IC50 = 800 nM T86702 CHXE26 44359791 IC50 = 200 nM T86702 C7VI5F 44359792 IC50 = 20 nM T86702 CAI78D 44359808 IC50 = 3000 nM T86702 CN0BH2 44359811 IC50 = 200 nM T86702 CYL4P0 44359813 IC50 = 20 nM T86702 CO7LW8 44359868 IC50 = 50 nM T86702 CAK2S0 44359869 IC50 = 300 nM T86702 CX9J2G 44359888 IC50 = 20 nM T86702 CU9I5B 44359889 IC50 = 2000 nM T86702 CLZG86 44359923 IC50 = 500 nM T86702 CF0P9S 44359924 IC50 = 2000 nM T86702 CIL92Y 44359925 IC50 = 200 nM T86702 CR35WH 44359926 IC50 = 500 nM T86702 CK6MD8 44360002 IC50 = 400 nM T86702 CL4F1H 44360016 IC50 = 500 nM T86702 CRW61Q 44360082 IC50 = 100 nM T86702 C9XZQ3 44360104 IC50 = 300 nM T86702 C4PF0M 44360162 IC50 = 5000 nM T86702 CQ60YD 44360219 IC50 = 25 nM T86702 CT4C6P 44360260 IC50 = 31 nM T86702 CY5I3O 44360286 IC50 = 46 nM T86702 C40OCB 44360287 IC50 = 1 nM T86702 C3IW9L 44360784 IC50 = 3.3 nM T86702 C90CYD 44367175 IC50 = 20 nM T86702 C2DV0R 44367276 IC50 = 11 nM T86702 C5BAW2 44367284 IC50 = 6 nM T86702 C2YG5E 44367285 IC50 = 222 nM T86702 CUDF82 44367309 IC50 = 21 nM T86702 CA0CJ1 44368580 IC50 = 570 nM T86702 CW0Y3K 44368632 IC50 = 478.63 nM T86702 CU8FD2 44368650 IC50 = 25 nM T86702 CLE71V 44368654 IC50 = 21.88 nM T86702 CQ27XL 44368655 IC50 = 72.44 nM T86702 CH9G3O 44368849 IC50 = 12.88 nM T86702 CV6ZG4 44368850 IC50 = 19 nM T86702 CB2U9G 44368858 IC50 = 10 nM T86702 CN78UB 44368864 IC50 = 20.89 nM T86702 CV8ZA4 44368865 IC50 = 6.761 nM T86702 CW8O3S 44368924 IC50 = 2818.38 nM T86702 C6CD9A 44368928 IC50 > 10000 nM T86702 C5HF6P 44368940 IC50 = 5000 nM T86702 CE30XV 44368941 IC50 = 2800 nM T86702 CG2P9T 44368942 IC50 = 10000 nM T86702 C7HT1U 44368944 IC50 = 3235.94 nM T86702 C1CW5A 44368946 IC50 = 8500 nM T86702 CV86QS 44368963 IC50 = 5011.87 nM T86702 C4C7UJ 44368968 IC50 = 562.34 nM T86702 C3EW6B 44368969 IC50 = 48 nM T86702 C4I6ME 44368970 IC50 = 8.913 nM T86702 C8IZC4 44369030 IC50 = 625 nM T86702 CDW8V9 44369031 IC50 = 275.42 nM T86702 C82BOI 44369038 IC50 > 10000 nM T86702 C65FBJ 44369041 IC50 = 3400 nM T86702 CI0S2R 44369094 IC50 = 8.71 nM T86702 CFI10T 44369095 IC50 = 2.57 nM T86702 CQGM80 44369096 IC50 = 25.7 nM T86702 CIR84S 44369104 IC50 = 120 nM T86702 C6SBW5 44369107 IC50 = 25 nM T86702 CAF5P0 44369163 IC50 = 770 nM T86702 CHC71X 44369164 IC50 = 110 nM T86702 CY5L0D 44369186 IC50 = 0.5 nM T86702 C1JZK6 44369209 IC50 = 39.81 nM T86702 C9BAO2 44369213 IC50 = 446.68 nM T86702 CCJ63B 44369214 IC50 = 3.8 nM T86702 C4E7DM 44369266 IC50 = 10 nM T86702 C92OKS 44369679 Ki = 30 nM T86702 C63WRQ 44369680 Ki > 650 nM T86702 CHV7Z8 44369681 Ki = 29.4 nM T86702 CX4ZU6 44369702 Ki > 650 nM T86702 C8ZK2I 44369876 Ki = 47.5 nM T86702 CI0ZD9 44371783 IC50 = 2490 nM T86702 C4VR5M 44371799 IC50 = 6150 nM T86702 C4FHG7 44371800 IC50 = 3795 nM T86702 C1QWA3 44374051 IC50 = 631 nM T86702 CX01WF 44374220 IC50 = 4084 nM T86702 C40TSF 44374235 IC50 = 4705 nM T86702 C1I6QU 44374342 IC50 = 3570 nM T86702 CZYL14 44374353 IC50 = 965 nM T86702 CGK04Y 44374370 IC50 = 7877 nM T86702 CCZ6J3 44379232 Ki = 3600 nM T86702 CW20ML 44379249 Ki = 9.5 nM T86702 CXM06G 44379250 Ki = 0.36 nM T86702 CK0B1D 44379273 Ki = 140 nM T86702 COD6P1 44379499 Ki = 1.9 nM T86702 C84YPO 44379547 Ki = 5800 nM T86702 C4M3CU 44380421 Ki = 32 nM T86702 C0CH2Q 44380422 Ki = 13 nM T86702 CBLY46 44380446 Ki = 25 nM T86702 C0F6ZP 44380458 Ki = 526 nM T86702 C1VY9Q 44380628 Ki = 7 nM T86702 C4H8SW 44380647 Ki = 100 nM T86702 CY03NT 44380706 Ki = 103 nM T86702 CHN0R1 44380983 Ki > 10000 nM T86702 CJ5W2S 44381004 Ki = 168 nM T86702 C82UHB 44381005 Ki = 28 nM T86702 C5A6EJ 44381025 Ki > 10000 nM T86702 C8A9FK 44381033 Ki = 13 nM T86702 C8D4SW 44381055 Ki > 10000 nM T86702 C3LIF2 44381197 Ki = 70 nM T86702 C27DGC 44381207 Ki = 13 nM T86702 C70VDN 44381208 Ki = 24 nM T86702 CMCN65 44383696 IC50 = 700 nM T86702 CYE90S 44383704 Ki = 82.4 nM T86702 C4O9DP 44383747 Ki = 0.53 nM T86702 C0W2SV 44383786 Ki = 0.5 nM T86702 C2UNW6 44383789 Ki = 2.95 nM T86702 C6V9FQ 44383801 Ki = 8.15 nM T86702 CV8UX5 44383829 Ki = 4.85 nM T86702 CCY30B 44383847 Ki = 12.8 nM T86702 C7MLD8 44383849 Ki = 2.43 nM T86702 C9F5LS 44384003 Ki = 67 nM T86702 CSM3P7 44384004 Ki = 162 nM T86702 CO9LJ6 44384005 Ki = 190 nM T86702 CJ4NV9 44384173 Ki = 47.8 nM T86702 C7B3AN 44384343 Ki = 12.3 nM T86702 C4B9NU 44384357 Ki = 51.4 nM T86702 CC81JP 44384395 Ki = 2.04 nM T86702 CKG95Y 44384455 Ki = 527 nM T86702 C96PAY 44384542 Ki = 6.41 nM T86702 C7HA0F 44384590 Ki = 64.4 nM T86702 C5ZYN1 44384591 Ki = 72.9 nM T86702 CVZ42A 44384592 Ki = 29.7 nM T86702 CSV63O 44384594 IC50 = 700 nM T86702 C49TAV 44384649 Ki = 34.9 nM T86702 CALI01 44384650 Ki = 5.43 nM T86702 C8SCB5 44384659 Ki > 650 nM T86702 C7A2HC 44384755 Ki = 14.9 nM T86702 CL51XE 44384756 Ki = 5.2 nM T86702 CD2PM4 44384761 Ki = 4.36 nM T86702 CJH8P4 44384762 Ki = 29.6 nM T86702 CH3M5X 44384813 Ki = 24.4 nM T86702 C59NBH 44384814 Ki = 5.19 nM T86702 C3EV2A 44384940 IC50 = 1000 nM T86702 C5AE0O 44384972 Ki = 11.6 nM T86702 CK7RP9 44385344 Ki = 24 nM T86702 CZ6PU7 44389401 Ki = 110 nM T86702 CO4W0Y 44389552 Ki = 430 nM T86702 CNPO26 44390575 IC50 = 500 nM T86702 CZB81D 44395506 IC50 = 3 nM T86702 CWGQ46 44404503 IC50 = 442 nM T86702 CLXM58 44404504 IC50 = 561 nM T86702 C0G4MR 44405997 IC50 > 380000 nM T86702 CZ0XC1 44405998 IC50 = 380000 nM T86702 C1F0DR 44406571 IC50 = 20 nM T86702 CHM26J 44406652 Ki = 2900 nM T86702 C1K3QM 44406655 IC50 = 500 nM T86702 C6YG5S 44406678 IC50 > 1000 nM T86702 C84ZSL 44411052 Ki = 12 nM T86702 CUE29K 44411053 Ki = 187 nM T86702 C6IKL1 44411602 IC50 = 28 nM T86702 CEB0S4 44411823 IC50 = 34 nM T86702 CT5PC9 44422672 IC50 = 45 nM T86702 CS9D5U 44422720 IC50 = 12 nM T86702 CNWM05 44422723 IC50 = 36 nM T86702 C58LAY 44422724 IC50 = 150 nM T86702 CDQU41 44422736 IC50 = 1200 nM T86702 CVUB56 44422737 IC50 = 440 nM T86702 CB8G2W 44422743 IC50 = 230 nM T86702 CK5H7O 44429877 IC50 = 1500 nM T86702 CWU7G8 44434565 IC50 > 100000 nM T86702 CF9HU5 44434566 IC50 = 1920 nM T86702 CV3M6F 44434578 IC50 = 21000 nM T86702 CJN1K9 44439853 Ki > 4500 nM T86702 CV58YW 44441018 Ki > 4501 nM T86702 CV85PN 44441019 Ki > 4501 nM T86702 C5O2WK 44441020 Ki > 4501 nM T86702 CU67WS 44441021 Ki > 4501 nM T86702 CXZ53B 44441022 Ki > 4501 nM T86702 C8S7UT 44441023 Ki > 4501 nM T86702 CT4PZ9 44441024 Ki > 4501 nM T86702 CU9GE6 44441025 Ki > 4501 nM T86702 CB2IT4 44441026 Ki > 4501 nM T86702 CN4X2F 44441027 Ki > 4501 nM T86702 CPF45Y 44441028 Ki > 4501 nM T86702 CAM23N 44441029 Ki > 4501 nM T86702 C23BPG 44441030 Ki > 4501 nM T86702 C5YMT6 44441031 Ki > 4501 nM T86702 C9A6GJ 44441032 Ki > 4501 nM T86702 CYSU19 44441033 Ki > 4501 nM T86702 C49CKM 44445388 IC50 = 164 nM T86702 CC2HV6 44445389 IC50 = 174 nM T86702 CWQ81G 44445390 IC50 = 161 nM T86702 C0HXS4 44445391 IC50 = 55 nM T86702 CT1CP7 44445392 IC50 = 420 nM T86702 CRNK10 44445393 IC50 = 960 nM T86702 CF0LR3 44445394 IC50 = 4 nM T86702 CH2Y7W 44445813 Ki = 36 nM T86702 C4J2QM 44445814 Ki = 218.78 nM T86702 C20HIJ 44446753 IC50 = 359 nM T86702 C4K5QT 44446756 IC50 = 4999 nM T86702 C47SRV 44446758 IC50 > 5000 nM T86702 C8HM5N 44446763 IC50 = 3500 nM T86702 CU5Z4V 44446765 IC50 > 5000 nM T86702 CYO65B 44446797 IC50 > 1000 nM T86702 CTKX08 44446807 IC50 > 5000 nM T86702 CJ1MP7 44446808 IC50 > 5000 nM T86702 CJN1L7 44446821 IC50 = 4000 nM T86702 C9FG5A 44446823 IC50 = 2601 nM T86702 C1P0BV 44446824 IC50 = 1669 nM T86702 C5AW3N 44446825 IC50 > 5000 nM T86702 C17YSI 44446827 IC50 > 5000 nM T86702 CE2OM1 44446839 IC50 = 4000 nM T86702 C49VJF 44446842 IC50 > 5000 nM T86702 CF4DL2 44446843 IC50 > 3000 nM T86702 CM7JV0 44447353 IC50 = 925 nM T86702 CSKN69 44455242 IC50 = 62.9 nM T86702 C3J1SV 44455676 IC50 = 964 nM T86702 C38VBL 44455836 IC50 = 308 nM T86702 CD9N5I 44459425 Ki = 118 nM T86702 CP98IX 44459426 Ki = 15 nM T86702 CAM2Q6 44459443 Ki = 99 nM T86702 CVY7O1 44460358 Ki = 229.09 nM T86702 C78GOL 44460359 Ki = 1584.89 nM T86702 C4MK3N 44460370 Ki = 330 nM T86702 CEY4L1 44460381 Ki > 10000 nM T86702 CEN93Y 44460382 Ki > 10000 nM T86702 CL30OP 44460588 Ki = 190 nM T86702 CO12NF 44460595 Ki = 109.65 nM T86702 C34BMW 44460598 Ki = 1778.28 nM T86702 C0A1KH 44460605 Ki = 190 nM T86702 CDN1V6 44460606 Ki = 830 nM T86702 C8TB4H 44460611 Ki > 10000 nM T86702 CJ6PN3 44460646 Ki = 42.66 nM T86702 CU8A1O 44460672 Ki = 1778.28 nM T86702 CIQ87B 44460676 Ki > 10000 nM T86702 C5B8NZ 44460690 Ki = 72 nM T86702 CK4WU2 44460737 Ki = 177.83 nM T86702 CY6JC5 44460927 Ki = 218.78 nM T86702 CG0Z7I 44478924 IC50 = 22000 nM T86702 CFO27Y 44478926 IC50 = 730 nM T86702 CBZJ29 44478927 IC50 = 1600 nM T86702 CRJ24K 44479197 IC50 = 1400 nM T86702 CGOH82 44479198 IC50 > 10000 nM T86702 CLV56M 44479199 IC50 = 7500 nM T86702 CY92OQ 44479458 IC50 = 60000 nM T86702 CH1QG9 44479459 IC50 = 4000 nM T86702 CB1NT7 44479460 IC50 = 23000 nM T86702 C0JQ9L 44479699 IC50 = 5600 nM T86702 C0DN1Q 44479700 IC50 > 100000 nM T86702 CTG24W 44479702 IC50 > 100000 nM T86702 CGZ49M 44479703 IC50 = 8000 nM T86702 CJ2BU5 44563487 IC50 = 1400 nM T86702 CP54WT 44563489 IC50 = 2538 nM T86702 C1UXP6 44563490 IC50 = 3863 nM T86702 CZ0W1A 44563491 IC50 = 174 nM T86702 C37UAM 44563492 IC50 = 463 nM T86702 C4BD0N 44563493 IC50 = 53 nM T86702 C7GF9S 44577362 IC50 = 330 nM T86702 CPT42K 44580109 IC50 > 5000 nM T86702 CQ7W5I 44580110 Ki > 4500 nM T86702 CQ4ZR1 44580422 IC50 = 2.1 nM T86702 CK68GT 44580539 Ki = 484 nM T86702 CXIY57 44580801 Ki > 10000000 nM T86702 C0OA8Y 44580802 Ki > 10000000 nM T86702 CNC4D7 44581071 Ki = 952000 nM T86702 CDF48U 44581111 Ki > 10000000 nM T86702 C2Z4HB 44583600 IC50 = 4999 nM T86702 C7PR8I 44583623 IC50 > 5000 nM T86702 CDRC42 44583654 IC50 > 5000 nM T86702 CM79HD 44583656 IC50 > 5000 nM T86702 CM9IN6 44592481 IC50 = 13300 nM T86702 CQFR57 44592482 IC50 = 13900 nM T86702 C19LWR 44634267 IC50 = 20 nM T86702 CM0I4J 45101511 IC50 = 5000 nM T86702 CACH13 45269631 IC50 = 920 nM T86702 CMPE63 45482676 IC50 = 54000 nM T86702 C4ZWY7 45487310 IC50 = 5000 nM T86702 C9SV0H 45487311 IC50 = 5000 nM T86702 CCF05Q 45487333 IC50 > 5000 nM T86702 CY09ZU 45487335 IC50 = 5000 nM T86702 COX40Y 45487358 IC50 > 5000 nM T86702 CF1T7M 45487359 IC50 = 5000 nM T86702 CRXI29 45487373 IC50 > 5000 nM T86702 CYL32E 45487376 IC50 > 5000 nM T86702 CO5P9I 45487386 IC50 > 5000 nM T86702 CS9Y8G 45487387 IC50 > 5000 nM T86702 CWLC18 45487393 IC50 > 5000 nM T86702 CI4KJ5 45487400 IC50 > 5000 nM T86702 C49HOI 45487401 IC50 = 5000 nM T86702 CSX5I9 46175170 IC50 = 68 nM T86702 CP8NT9 46225509 Ki > 10000 nM T86702 C8HX7K 46840956 IC50 = 74340 nM T86702 CH0Z1E 46844314 Ki > 40000 nM T86702 C5L8GF 46871738 IC50 = 300 nM T86702 CR1KF7 46871739 IC50 = 130 nM T86702 C8Q6YR 46871740 IC50 = 24.5 nM T86702 C58YSM 46871741 IC50 = 160 nM T86702 C3X5EN 46873064 IC50 = 87770 nM T86702 C0S9WB 46919610 Ki = 19000 nM T86702 CUD7O0 50941549 IC50 = 9600 nM T86702 CU2SX3 51355576 Ki > 10000 nM T86702 CLA96C 53232689 Ki = 3 nM T86702 C3BGW0 53233015 Ki > 40000 nM T86702 CTQ02K 53320639 IC50 = 3900 nM T86702 C4UE6R 53322469 IC50 > 100000 nM T86702 CZD9L1 53324788 IC50 = 8960 nM T86702 CPY02U 53327890 IC50 = 180 nM T86702 CPGE80 53327891 IC50 = 93 nM T86702 CLJ4G2 53328858 IC50 = 46 nM T86702 C4G3QL 53328859 IC50 = 38 nM T86702 CX1TW0 53328860 IC50 = 11 nM T86702 C0ZX5G 53329215 IC50 = 84 nM T86702 CSU52A 53329216 IC50 = 320 nM T86702 CNB63X 53361475 IC50 = 12100 nM T86702 C6Y2EV 53374826 IC50 > 100000 nM T86702 C3LF0P 54580544 Ki = 130 nM T86702 C6R3MZ 54580973 Ki > 50000 nM T86702 CVO09J 54581546 Ki = 44 nM T86702 CWKA42 54582019 Ki > 50000 nM T86702 CD09BZ 54582543 IC50 = 90 nM T86702 CK52YD 54583511 Ki = 59 nM T86702 CG37UX 54587429 Ki = 9.9 nM T86702 CL9SC3 54587769 Ki > 40000 nM T86702 C13FSJ 54669762 Ki = 23400 nM T86702 CHS01Z 54669766 Ki = 40500 nM T86702 CC67RV 54681831 IC50 = 10 nM T86702 CEP48O 54685358 IC50 = 2400 nM T86702 C83NUI 54687474 IC50 = 240 nM T86702 CZ6V0U 54724681 IC50 = 19 nM T86702 CJ6HT4 54726662 IC50 = 16400 nM T86702 CAEV82 54726663 IC50 = 3700 nM T86702 C9P5ES 54752445 IC50 = 90 nM T86702 C0HKC9 54752446 IC50 = 86 nM T86702 C62FZC 56835063 IC50 = 2530 nM T86702 CKJ9S1 56835167 IC50 = 220 nM T86702 C21CLZ 56835168 IC50 = 3900 nM T86702 C0L2TS 56835169 IC50 = 3400 nM T86702 CHE2I1 57345500 Ki > 50000 nM T86702 C63TFM 57345501 Ki > 50000 nM T86702 C8KT2F 57345502 Ki = 31000 nM T86702 C0KPD8 57384084 IC50 = 2000 nM T86702 CV67JB 57384091 IC50 = 4000 nM T86702 CR8MW2 57391205 IC50 > 10000 nM T86702 CP5BX6 57394607 IC50 = 493 nM T86702 CNOH63 57394711 IC50 > 10000 nM T86702 CE5X3D 57394850 IC50 = 700 nM T86702 CG43ME 57394903 IC50 = 160 nM T86702 CWH7V8 57561293 IC50 = 5500 nM T86702 CY1N3J 57792153 IC50 = 1082 nM T86702 CCKD80 58307579 Ki = 350 nM T86702 C5AQG2 68724898 Ki > 10000 nM T86702 CHL56C 68799256 Ki > 10000 nM T86702 CT2K3G 70265758 Ki = 7210 nM T86702 CHRO48 70266605 Ki > 10000 nM T86702 C34LYX 70266607 Ki > 10000 nM T86702 COD03W 70267879 Ki > 10000 nM T86702 CG38ZM 70267887 Ki > 10000 nM T86702 C50CAL 70268171 Ki = 8730 nM T86702 CWP71E 70269104 Ki > 10000 nM T86702 CGD3B2 70269997 Ki > 10000 nM T86702 CH76IU 70684364 Ki = 27000 nM T86702 CZ63AG 70684365 Ki = 17000 nM T86702 C8B6WD 70688393 IC50 = 8150 nM T86702 CGR3J2 70688394 IC50 = 22300 nM T86702 C3LCG0 70688633 Ki = 12000 nM T86702 C6P3XM 70693710 Ki > 50000 nM T86702 C0HE2P 70694634 IC50 = 14810 nM T86702 CGCM02 71454432 IC50 = 10000 nM T86702 CYB60V 71458014 IC50 = 230 nM T86702 CKW27N 71461578 IC50 = 910 nM T86702 CH5J4A 71602247 IC50 = 7100 nM T86702 CH53IU 71602248 IC50 = 67000 nM T86702 C97EWQ 71602249 IC50 = 6800 nM T86702 CYS46I 71652677 IC50 = 4000 nM T86702 CX67VE 71654516 IC50 = 3400 nM T86702 C6KEH0 71680708 Ki = 2500 nM T86702 C7DMX5 71680709 Ki = 460 nM T86702 CFPM82 71680710 Ki = 37 nM T86702 C9ZOM7 71680866 Ki = 2000 nM T86702 CQ68LT 71680868 Ki > 100000 nM T86702 CFH2V0 71681183 Ki = 1600 nM T86702 CV3X1T 71682766 Ki > 200000 nM T86702 C80EYX 71682913 Ki > 200000 nM T86702 CIBD03 71682914 Ki = 10000 nM T86702 C41BYG 71682915 Ki > 200000 nM T86702 C93XEI 71682916 Ki = 100000 nM T86702 CQ29PJ 71682917 Ki > 200000 nM T86702 CFWN65 71683062 Ki > 200000 nM T86702 C61NKZ 72720906 IC50 = 21 nM T86702 C7XWM5 72948626 IC50 = 10 nM T86702 CR70EY 72948808 IC50 = 9 nM T86702 C2WV4D 72948991 IC50 = 7270 nM T86702 CA76TR 72948995 IC50 = 15 nM T86702 CZ95GN 72949172 IC50 = 6 nM T86702 C38IDL 73345835 Ki = 1.9 nM T86702 CE05UK 73347034 Ki > 10000 nM T86702 C9W7OB 73348532 Ki = 1600 nM T86702 CW01EA 73349535 IC50 > 10000 nM T86702 C8ROG3 73350414 Ki = 990 nM T86702 CF7AB2 73350415 Ki = 300 nM T86702 C2PFM4 73351930 Ki = 4100 nM T86702 CC7OE8 73354605 Ki = 1300 nM T86702 CX6S3Y 73354606 Ki = 540 nM T86702 CGS1Q4 73354607 IC50 = 19000 nM T86702 C4X9OZ 73354608 Ki = 5300 nM T86702 CI09CY 73354906 Ki = 31 nM T86702 CA5T7P 73603957 IC50 = 15000 nM T86702 C8VN1R 74221194 IC50 = 2800 nM T86702 CUB7V9 76329513 IC50 = 4.2 nM T86702 CUE7G4 86287514 IC50 = 50000 nM T86702 CGQ8F3 86287515 IC50 = 1900 nM T86702 CJ37XE 86287516 IC50 = 23000 nM T86702 COV8I9 86291010 IC50 = 1020 nM T86702 CSH7A5 90033597 IC50 = 18900 nM T86702 CO2FL5 90137145 IC50 = 660 nM T86702 CYZP25 91824169 IC50 > 10000 nM T86702 CRT54C 101910871 IC50 = 69000 nM T86702 C0M3QS 118179775 IC50 = 21 nM T86702 C0XML2 118179776 IC50 = 16 nM T86702 C0W3NG 118179777 IC50 = 476 nM T86702 CX9YG0 118179779 IC50 = 6 nM T86702 CW1TU9 118179786 IC50 = 46 nM T86702 CRG2W5 118179799 IC50 = 178 nM T86702 CH35NR 118179800 IC50 = 5 nM T86702 CK54UB 118179801 IC50 = 916 nM T86702 CP8QO0 118179807 IC50 = 19 nM T86702 CT4G5D 118179817 IC50 = 39 nM T86702 CIU02H 118179819 IC50 = 4 nM T86702 CD9TG2 118179830 IC50 = 132 nM T86702 CN72KV 118179833 IC50 = 114 nM T86702 CZ01AH 118179837 IC50 = 314 nM T86702 C6TR4O 118179845 IC50 = 20000 nM T86702 C5TZ1D 118179847 IC50 = 7 nM T86702 CVWR97 118179850 IC50 = 38600 nM T86702 CT8U1K 118179865 IC50 = 9600 nM T86702 CR64FW 118179867 IC50 = 96 nM T86702 CIXQ34 118179870 IC50 = 4 nM T86702 C27XIK 118225133 IC50 > 10000 nM T86702 C58KIN 118233723 IC50 > 10000 nM T86702 CU6ES2 118233724 IC50 > 10000 nM T86702 C8ET1Z 118233725 IC50 > 10000 nM T86702 C9P0LC 118233726 IC50 > 10000 nM T86702 C8SIM0 118233727 IC50 > 10000 nM T86702 CQTE52 118233728 IC50 > 10000 nM T86702 CEVI64 118233730 IC50 > 10000 nM T86702 C08CPE 118233731 IC50 > 10000 nM T86702 C8Q5XC 118233733 IC50 > 10000 nM T86702 CZQO42 118233734 IC50 > 10000 nM T86702 CCDG68 118233743 IC50 > 10000 nM T86702 C25TYU 118233744 IC50 > 10000 nM T86702 CL5UV6 118233745 IC50 > 10000 nM T86702 C8XWB9 118233746 IC50 > 10000 nM T86702 CC7K9R 118233747 IC50 > 10000 nM T86702 CGA7J1 118233748 IC50 > 10000 nM T86702 CVIG81 118233749 IC50 > 10000 nM T86702 CTU81Y 118233750 IC50 > 10000 nM T86702 CCA6W2 118233751 IC50 > 10000 nM T86702 C60QIZ 118233752 IC50 > 10000 nM T86702 CS5G9T 118233753 IC50 > 10000 nM T86702 C5ZS4E 118722686 IC50 = 3000 nM T86702 CIZB24 118722687 IC50 = 20000 nM T86702 C5C0ZX 118722688 IC50 = 64000 nM T86702 CGKD16 118734983 IC50 = 20 nM T86702 C84NEC 118734984 IC50 = 65 nM T86702 CX7H5Q 118734985 IC50 = 18 nM T86702 CH6OW5 122179777 IC50 = 82560 nM T86702 CH1GT7 123144081 IC50 > 10000 nM T86702 C9QKI3 127020966 IC50 > 100000 nM T86702 CPG8E6 127027350 Ki > 10000 nM T86702 CXS26T 127027351 Ki > 10000 nM T86702 C52FZR 127028674 IC50 = 130000 nM T86702 CR19OH 127028675 IC50 = 15000 nM T86702 C8KE7R 127028996 IC50 = 45000 nM T86702 CYA92R 130282633 IC50 = 90 nM T86702 CO3QE2 130282636 IC50 = 90 nM T86702 CTN42D 132941363 IC50 = 60000 nM T86702 CTS0G5 132967549 IC50 = 100000 nM T86702 CJP4B3 132967551 IC50 = 10000 nM T86702 CS3YZ1 132967554 IC50 = 150000 nM T86702 CHV2U1 135438561 IC50 = 4000 nM T86702 CJ7Z3R 135454124 IC50 = 31000 nM T86702 C4FVJ1 135487604 IC50 = 78000 nM T86702 C29AGZ 136036767 IC50 = 5060 nM T86702 CMXL16 136036768 IC50 = 65000 nM T86702 C8WP2X 136036769 IC50 >= 100000 nM T86702 CO19FB 136036770 IC50 = 6190 nM T86702 CQS0B6 136036777 IC50 >= 100000 nM T86702 CU5IK0 136036779 IC50 = 43000 nM T86702 C49YHB 136036783 IC50 = 3150 nM T86702 CU54MP 136036786 IC50 = 10350 nM T86702 C12UID 136036787 IC50 >= 100000 nM T86702 CA5JR6 136054481 IC50 = 370 nM T86702 CV47JN 136054485 IC50 = 23 nM T86702 CZ48WO 136054487 IC50 = 2400 nM T86702 C8FGT0 136054495 IC50 = 3300 nM T86702 CG70BZ 136054516 IC50 = 2.5 nM T86702 CSM57W 136054520 IC50 = 2.6 nM T86702 CXNG40 136118011 Ki = 567 nM T86702 C1IOH9 136118012 Ki > 4501 nM T86702 CJG54U 136219136 IC50 > 30000 nM T86702 C3CAV5 136219141 IC50 > 30000 nM T86702 CPB07Z 136241630 IC50 = 6400 nM T86702 CIEW62 136380958 IC50 = 30 nM T86702 CHOA14 136814721 IC50 >= 100000 nM T86702 CFJ3I6 136814723 IC50 = 97350 nM T86702 C9HS7J 137287436 IC50 = 1.5 nM T86702 C0I6RH 137632487 IC50 = 4.3 nM T86702 CB8M6U 137646865 IC50 = 4400 nM T86702 CS80YI 137652598 IC50 = 2000 nM T86702 CAB7Q6 137660566 IC50 > 10000 nM T86702 CZ8H6N 137661550 IC50 = 17000 nM T86702 CYFQ54 144883303 IC50 > 10000 nM T86702 CA2EI4 144883305 IC50 > 10000 nM T86702 CX80ML 144883318 IC50 > 10000 nM T86702 CQYH92 145949456 IC50 > 10000 nM T86702 C2SM0T 145950300 IC50 > 10000 nM T86702 C85BXD 145951133 IC50 > 10000 nM T86702 C6JP8O 145955500 IC50 > 10000 nM T86702 CXT3I5 145958912 IC50 > 10000 nM T86702 CQN59P 145959729 IC50 > 10000 nM T86702 CX6R5D 145959924 IC50 > 10000 nM T86702 C8UC1T 145963891 IC50 = 52800 nM T86702 CWOF29 145964116 IC50 = 47200 nM T86702 CKD86B 145964366 IC50 = 30200 nM T86702 CI0T9C 145964617 IC50 = 35300 nM T86702 C3MDU9 145965508 IC50 = 40930 nM T86702 CA94UB 145966060 IC50 = 10200 nM T86702 CL7QD9 145966162 IC50 = 21300 nM T86702 CA80DF 145966420 IC50 = 40800 nM T86702 CNR98O 145966867 IC50 = 28000 nM T86702 CI9JB5 145967177 IC50 = 39700 nM T86702 CJ47BV 145969859 IC50 = 22600 nM T86702 C1R9ES 145971386 IC50 = 6700 nM T86702 CQ78MP 145971807 IC50 > 100000 nM T86702 CX0JY3 145972073 IC50 > 100000 nM T86702 C0K4JW 145972664 IC50 > 10000 nM T86702 CPB91X 145972781 IC50 = 400 nM T86702 CQ4K0X 145972990 IC50 > 100000 nM T86702 CG4E3F 145973485 IC50 = 12800 nM T86702 CTA0S4 145974193 IC50 = 8800 nM T86702 C52HKA 145974836 IC50 = 23800 nM T86702 CKW8B6 145975533 IC50 = 25500 nM T86702 CV9D1F 145975682 IC50 > 100000 nM T86702 CTD40B 145975699 IC50 > 100000 nM T86702 CMNS71 145975707 IC50 = 1000 nM T86702 CM6QB0 145976230 IC50 > 100000 nM T86702 CU7HO6 145976282 IC50 = 24900 nM T86702 CW6F2Y 145976412 IC50 = 19600 nM T86702 C5C6VJ 145976464 IC50 = 66120 nM T86702 CBD28P 145977013 IC50 = 59700 nM T86702 C8CV6O 145977231 IC50 > 100000 nM T86702 C3VOQ8 145978127 IC50 = 26900 nM T86702 C2JQ6E 145978441 IC50 = 21500 nM T86702 C8ZVJ6 145978450 IC50 = 58300 nM T86702 C42JOA 145978615 IC50 > 100000 nM T86702 CZ25LW 155512044 IC50 = 51000 nM T86702 CP9YX2 155567218 IC50 = 7100 nM T86702 CU42CE 155567829 IC50 > 100000 nM T86702 C8D5VK 155567855 IC50 = 23000 nM T86702 CV4TJ8 11794277 Ki = 330 nM T86702 D01BCK 23382 IC50 = 50000 nM T86702 D02ECA 448942 IC50 = 390 nM T86702 D02EFQ 10549609 IC50 = 8 nM T86702 D02UYR 9907830 Ki = 15.2 nM T86702 D03MUZ 17759555 IC50 = 2300 nM T86702 D03WJG 9910222 Ki = 0.51 nM T86702 D04GOO 10111838 IC50 > 100000 nM T86702 D04VPH 45376872 IC50 > 22000 nM T86702 D05THD 44478925 IC50 = 45000 nM T86702 D06EHW 11625778 IC50 = 3560 nM T86702 D07DRT 46175162 Ki = 810 nM T86702 D07GEL 10344307 Ki = 14 nM T86702 D07MJD 44479701 IC50 = 74000 nM T86702 D08CBB 9060 IC50 > 500000 nM T86702 D09EUH 9819306 IC50 < 1000 nM T86702 D09ZOA 25049753 IC50 = 320 nM T86702 D0A0FY 44479457 IC50 > 50000 nM T86702 D0A4TC 446504 IC50 = 14 nM T86702 D0B3UN 44580458 Ki = 40 nM T86702 D0BI8T 44288042 IC50 = 0.8 nM T86702 D0D7UA 10267279 IC50 = 500 nM T86702 D0F7BE 4369084 Ki = 707.95 nM T86702 D0G3YZ 11391583 IC50 > 98000 nM T86702 D0H2PA 9886977 Ki = 0.9 nM T86702 D0H6CK 10160968 Ki = 91 nM T86702 D0J5EZ 54726664 IC50 = 5600 nM T86702 D0K4TI 49292 IC50 = 30000 nM T86702 D0N8YA 159596 IC50 > 100000 nM T86702 D0NP8A 10370504 IC50 = 5.9 nM T86702 D0OR6O 91623362 IC50 = 15 nM T86702 D0P2TS 9818682 IC50 > 10000 nM T86702 D0Q4TA 10044321 IC50 = 4500 nM T86702 D0R2BO 194777 IC50 = 43 nM T86702 D0S9OL 10155934 IC50 = 27000 nM T86702 D0T1FR 44457233 IC50 > 100000 nM T86702 D0W2UK 6914621 Ki = 141 nM T86702 D0W3ME 4369080 Ki = 18 nM T86702 D0XK7G 10445302 Ki = 4400 nM T86702 D0XL8K 44313734 IC50 = 160 nM T86702 D0Y5IQ 44255320 IC50 = 5000 nM T86702 D0Y7NV 2220392 IC50 = 9000 nM T78205 D00HGB 4488 IC50 = 149000 nM T78205 D05FTJ 4044 IC50 = 124000 nM T78205 D06ACW 6083 IC50 = 70000 nM T78205 D09GOS 2812 IC50 < 3000 nM T78205 D0B2WJ 3371 IC50 = 70000 nM T78205 D0EV8E 3198 IC50 < 3000 nM T78205 CKFN90 33576 EC50 = 100000 nM T78205 C0BE1A 85472 IC50 = 76000 nM T78205 CX4SM7 636430 IC50 = 100000 nM T78205 CYT5D3 9948349 IC50 = 600 nM T78205 C4K2OE 16219859 IC50 = 25 nM T78205 CI14ZM 21637538 IC50 = 210 nM T78205 CUG7J9 24814386 IC50 = 300000 nM T78205 CJ6EK2 76310334 IC50 = 15000 nM T78205 CNW38T 76314001 IC50 = 100000 nM T78205 C5QJ2Z 76314003 IC50 = 11000 nM T78205 CGMJ04 76321279 IC50 = 100000 nM T78205 C1BDL2 76321280 IC50 = 3000 nM T78205 CK5CY6 76328457 IC50 < 900000 nM T78205 C2LU7Z 76332138 IC50 = 51000 nM T78205 CLHZ25 76335751 IC50 = 49000 nM T78205 C3TW0A 134374895 IC50 > 30000 nM T78205 CEK6B1 139300630 IC50 > 10000 nM T78205 CW72XD 145951922 IC50 = 4600 nM T78205 C93RZI 145955484 IC50 = 5100 nM T78205 C40RXH 145957829 IC50 = 4000 nM T78205 CCQ19B 145972219 IC50 = 3700 nM T78205 D00HCI 1598 IC50 = 1000 nM T78205 D0N7MS 5353376 IC50 = 320 nM T88505 D07SDQ 969516 EC50 = 21000 nM T88505 D0JU5X 400769 EC50 = 60 nM T88505 D0U3EP 445154 EC50 = 5400 nM T88505 D04ILM 73053707 EC50 = 530 nM T88505 C7Z9YP 73432 IC50 = 29.19 nM T88505 C8Y7AX 641324 EC50 = 7200 nM T88505 C5TM3K 685506 EC50 > 10000 nM T88505 C7KVG3 830608 EC50 = 3300 nM T88505 CTU28L 839341 EC50 = 4700 nM T88505 C5V4UP 977560 EC50 = 3000 nM T88505 C9GOD0 1125827 EC50 = 10300 nM T88505 C5ZN1R 1551564 EC50 = 1040 nM T88505 C2GZ3U 1737815 EC50 = 8000 nM T88505 CH17LY 1811454 EC50 = 18100 nM T88505 CI87QD 5281396 EC50 = 1200 nM T88505 CR2NP0 5375540 EC50 = 12400 nM T88505 CHWE83 5375541 EC50 = 3100 nM T88505 CU7MX6 5375953 EC50 = 4400 nM T88505 CU6G8J 5472867 EC50 = 3300 nM T88505 CK2RN0 5708421 EC50 = 21100 nM T88505 C1A4LQ 5788151 EC50 > 100000 nM T88505 CT43WB 5816652 EC50 > 100000 nM T88505 CKFY48 5896779 EC50 = 93020 nM T88505 C0E3PX 5944124 EC50 > 100000 nM T88505 C59FHR 5951878 EC50 > 100000 nM T88505 C02UPR 5997893 EC50 = 1320 nM T88505 CUEK97 6036014 EC50 = 1480 nM T88505 C8LV9C 6258021 EC50 = 7600 nM T88505 CQ64LS 6537003 EC50 > 100000 nM T88505 CP1D0M 9952605 EC50 = 16600 nM T88505 CIB45A 10036098 EC50 = 1400 nM T88505 C6KBI5 10330812 EC50 = 1300 nM T88505 CK8VO6 10420716 EC50 = 800 nM T88505 COV54C 10553752 EC50 = 2450 nM T88505 CRKC63 10601247 EC50 > 25000 nM T88505 CA41EF 10673649 EC50 > 25000 nM T88505 CDS5X3 10688261 EC50 = 14400 nM T88505 C05NWT 10695622 EC50 > 25000 nM T88505 C2L3GK 10719972 EC50 > 25000 nM T88505 CTAP81 10743719 EC50 = 1097 nM T88505 CRF19I 10840295 EC50 = 11480 nM T88505 C8U0FG 11148621 EC50 = 650 nM T88505 CD8Z3I 11160198 EC50 = 11400 nM T88505 C7A0VY 11241653 EC50 = 4200 nM T88505 CQ21KF 11299420 EC50 = 3700 nM T88505 CBF80W 11379138 EC50 > 15000 nM T88505 CX58OF 11600967 EC50 = 4300 nM T88505 C8C3FZ 11746024 EC50 = 1000 nM T88505 CLR83A 11788847 EC50 = 700 nM T88505 C3ZG1M 11983527 EC50 = 7300 nM T88505 CW5G1P 12967780 EC50 > 25000 nM T88505 C25OTQ 15113696 EC50 = 1600 nM T88505 C01REY 15113698 EC50 = 5400 nM T88505 CM42PH 15270381 EC50 > 10000 nM T88505 C3GP0Q 15578704 EC50 = 3100 nM T88505 CKCD63 15863790 EC50 > 25000 nM T88505 CN76ZE 16737013 EC50 = 4600 nM T88505 CBF9G6 23233795 EC50 = 8900 nM T88505 C5SZL8 23652110 EC50 = 3700 nM T88505 C2JDN4 24420623 EC50 = 1778 nM T88505 CH3W2C 26946782 EC50 = 1334 nM T88505 C5EJB0 32737690 EC50 = 1155 nM T88505 CGP5B1 44563765 EC50 = 9500 nM T88505 C7BSA3 49799649 EC50 = 2600 nM T88505 C4ZT1B 66772006 EC50 = 4400 nM T88505 CGS4M5 66772015 EC50 = 3600 nM T88505 CI9T0W 66772172 EC50 > 15000 nM T88505 CYEM86 68372424 EC50 = 3300 nM T88505 C9TRM0 71508695 EC50 = 5300 nM T88505 C7R5EZ 71571581 EC50 = 8600 nM T88505 CLYU51 72189364 EC50 = 8659 nM T88505 C8VAE9 72189366 EC50 > 10000 nM T88505 COG8P7 72189368 EC50 > 10000 nM T88505 CJ9NR2 72189370 EC50 = 3230 nM T88505 CW5X0P 72190289 EC50 = 9070 nM T88505 C6EP9O 72190290 EC50 > 10000 nM T88505 CTN0R7 72190291 EC50 = 1517 nM T88505 C4DR6Y 72190292 EC50 = 849 nM T88505 CB2JF8 72190293 EC50 > 10000 nM T88505 CIU3Q8 72190294 EC50 = 178 nM T88505 C5HJC2 72190605 EC50 = 148 nM T88505 C1LB6C 72711039 EC50 > 100000 nM T88505 CRG72Q 72711263 EC50 > 100000 nM T88505 CK4JI9 72711264 EC50 > 100000 nM T88505 CNT4Z5 72711265 EC50 > 100000 nM T88505 CVFC95 72711266 EC50 > 100000 nM T88505 CI7WQ9 72711267 EC50 > 100000 nM T88505 CWG7B0 72711268 EC50 > 100000 nM T88505 C96SDP 72711269 EC50 > 100000 nM T88505 CR01FB 72711493 EC50 > 100000 nM T88505 CTY95W 72711494 EC50 > 100000 nM T88505 C69ZSY 72711495 EC50 > 100000 nM T88505 CUQB94 72711496 EC50 > 100000 nM T88505 C9VR5N 72711497 EC50 > 100000 nM T88505 CSJ0T7 72711498 EC50 > 100000 nM T88505 CVD46M 72711499 EC50 > 100000 nM T88505 CGPO82 72711731 EC50 > 100000 nM T88505 C3M5XL 72711732 EC50 > 100000 nM T88505 C4T3RL 72711733 EC50 = 87950 nM T88505 CF39YO 72711734 EC50 > 100000 nM T88505 CTI4X1 72711735 EC50 > 100000 nM T88505 C7C4HJ 72711736 EC50 = 75850 nM T88505 CR30NP 72711939 EC50 = 49610 nM T88505 C8VIT5 72711940 EC50 > 100000 nM T88505 CGH5S8 72711941 EC50 = 92000 nM T88505 CH5VW0 72711942 EC50 = 81540 nM T88505 CYGK50 72711943 EC50 = 58540 nM T88505 CQ0UD3 72711944 EC50 > 100000 nM T88505 CJD3E1 72712141 EC50 > 100000 nM T88505 CER0L2 72712142 EC50 > 100000 nM T88505 CEPI87 72712143 EC50 > 100000 nM T88505 CL65GX 72712144 EC50 > 100000 nM T88505 CH19AK 72712145 EC50 > 100000 nM T88505 C5K2SE 72712146 EC50 = 58860 nM T88505 CF73OT 72712147 EC50 = 59120 nM T88505 C4F3VH 73355399 EC50 > 100000 nM T88505 C4QEP1 76308437 EC50 > 15000 nM T88505 CLH89J 76326519 EC50 = 900 nM T88505 CU6E0X 90644814 EC50 = 3100 nM T88505 CL1Y7W 90666859 EC50 = 800 nM T88505 C9K8ZB 101161159 EC50 = 6900 nM T88505 C1PIQ2 101161160 EC50 = 1400 nM T88505 CYG4Q3 118169882 EC50 = 1600 nM T88505 CVX89N 118169940 EC50 = 83 nM T88505 CVT45P 118170010 EC50 = 760 nM T88505 CGP2N1 118170044 EC50 = 850 nM T88505 C1KYL6 118170387 EC50 = 11 nM T88505 CMW6L4 118170433 EC50 = 2900 nM T88505 C8R1EV 118170437 EC50 = 3400 nM T88505 CLN34U 118188783 EC50 = 570 nM T88505 C8QRI5 118370757 EC50 = 1500 nM T88505 CP9N7W 122190547 IC50 = 5390 nM T88505 C7U6SV 122653346 EC50 = 30 nM T88505 CP1SA8 122653376 EC50 = 1400 nM T88505 CA25XY 134132759 EC50 = 9600 nM T88505 CP61DX 134135915 EC50 = 2900 nM T88505 CT1P5Z 134137387 EC50 = 6000 nM T88505 C8E0MA 134138511 EC50 = 5100 nM T88505 CDO07A 134139310 EC50 = 2700 nM T88505 CGP6H4 134141818 IC50 = 115 nM T88505 C4N9KW 134141839 EC50 > 15000 nM T88505 CU8NW7 134143055 EC50 = 2600 nM T88505 CB07JR 134144207 EC50 = 3800 nM T88505 CJD9C5 134145422 EC50 = 1100 nM T88505 CN3IQ2 134145873 EC50 > 15000 nM T88505 CUR09F 134146382 EC50 = 5900 nM T88505 C9FDL0 134146522 EC50 = 3200 nM T88505 C0CNL7 134148569 EC50 = 300 nM T88505 CG0R3F 134149461 EC50 = 1900 nM T88505 CN1D3K 134152632 EC50 = 2000 nM T88505 CDE0P7 134153095 EC50 = 2900 nM T88505 CSWV05 134153135 EC50 = 2200 nM T88505 CUT3M5 134154604 EC50 > 15000 nM T88505 CJMU05 134154807 EC50 = 450 nM T88505 CI2R1Q 134155179 EC50 = 2300 nM T88505 COXF83 134155861 EC50 = 5000 nM T88505 C3J6IP 134157818 EC50 = 3100 nM T88505 C62RLG 145963983 EC50 > 25000 nM T88505 C2QVC5 145964968 EC50 > 25000 nM T88505 COGN67 145965850 EC50 > 25000 nM T88505 CTCE64 145965867 EC50 > 25000 nM T88505 C31UPV 145965989 EC50 > 25000 nM T88505 CI6CL4 145966660 EC50 > 25000 nM T88505 CP68JQ 145977608 EC50 > 25000 nM T88505 C1T5VP 146380951 EC50 = 908 nM T88505 CHD2X0 153404509 EC50 = 346 nM T88505 C34FVT 153404513 EC50 = 327 nM T88505 CL1KX6 153635800 EC50 = 1204 nM T88505 C1MQT9 155511967 EC50 > 10000 nM T88505 CAG9P8 155512898 EC50 = 2500 nM T88505 C7KMV9 155513109 EC50 = 948 nM T88505 C9YF1X 155513623 EC50 = 2642 nM T88505 C84EHX 155515902 EC50 > 10000 nM T88505 C4FD6M 155517566 EC50 = 165 nM T88505 CS2UI9 155517757 EC50 > 50000 nM T88505 C7KBT1 155518477 EC50 = 22800 nM T88505 CZM8N7 155518704 EC50 = 6350 nM T88505 C0B4XC 155519258 EC50 = 7383 nM T88505 CVP0Z3 155519471 EC50 = 29500 nM T88505 C09DKY 155520452 EC50 > 10000 nM T88505 C5VQS0 155524592 EC50 = 7021 nM T88505 CU90LV 155525158 EC50 = 347 nM T88505 CATG19 155525392 EC50 = 1198 nM T88505 C07YPO 155525419 EC50 > 10000 nM T88505 C34QPD 155526171 EC50 = 877 nM T88505 C6IJ2M 155526306 EC50 = 1083 nM T88505 CK98UF 155527259 EC50 = 955 nM T88505 CBON75 155527345 EC50 > 10000 nM T88505 CWC8E6 155528319 EC50 = 943 nM T88505 C60DWO 155528387 EC50 = 26300 nM T88505 CK07XG 155529092 EC50 = 3270 nM T88505 CA27QK 155529557 EC50 = 786 nM T88505 C5CBG6 155530050 EC50 > 10000 nM T88505 C2OG5B 155530251 EC50 = 1900 nM T88505 C1OX2C 155531540 EC50 = 6287 nM T88505 CZL2J7 155531909 EC50 = 202 nM T88505 CVH7Z8 155532575 EC50 = 1200 nM T88505 CHJ4N0 155533319 EC50 = 237 nM T88505 C9N3EY 155536526 EC50 = 246 nM T88505 CFYM47 155537393 EC50 > 50000 nM T88505 C1JTZ2 155537472 EC50 = 655 nM T88505 CS6WY2 155538727 EC50 = 17800 nM T88505 CM56QD 155539584 EC50 = 7978 nM T88505 C7XBH1 155541239 EC50 = 6312 nM T88505 C5OF9X 155543628 EC50 = 15500 nM T88505 CGE4J1 155543675 EC50 = 2171 nM T88505 CTMV94 155544022 EC50 = 698 nM T88505 CF84UT 155544070 EC50 = 5000 nM T88505 C78ARS 155545140 EC50 = 7610 nM T88505 CAEU17 155545372 EC50 = 124 nM T88505 CBIO03 155547371 EC50 > 50000 nM T88505 C7R3HE 155548228 EC50 = 16200 nM T88505 C0SB6J 155552871 EC50 > 10000 nM T88505 C8NKL3 155553157 EC50 = 6845 nM T88505 CY05NR 155554308 EC50 = 348 nM T88505 CBEY86 155556533 EC50 > 50000 nM T88505 CVK6D1 155556547 EC50 = 444 nM T88505 CVO9C6 155558557 EC50 > 10000 nM T88505 CM12ID 155559174 EC50 = 142 nM T88505 CF61CD 155559382 EC50 = 350 nM T88505 CN1U5F 155560023 EC50 = 1007 nM T88505 C3V4KN 155561540 EC50 > 10000 nM T88505 C62OSI 155561561 EC50 > 50000 nM T88505 C1E3IZ 155561727 EC50 = 1600 nM T88505 C1PCO9 155561916 EC50 = 9355 nM T88505 CCGO48 155562556 EC50 > 10000 nM T88505 C5Q9SZ 155563702 EC50 = 1155 nM T88505 C2TQS4 155564048 EC50 = 132 nM T88505 C5NVI2 155565186 EC50 > 50000 nM T88505 CL8HY9 155566001 EC50 > 50000 nM T88505 C8DGR5 155566478 EC50 = 76 nM T88505 C4MF7U 155566926 EC50 = 98 nM T88505 CB9O2T 155569050 EC50 = 16300 nM T88505 D0DQ2G 16043 EC50 = 91530 nM T88505 D0IO0I 6474893 EC50 = 900 nM T88505 D0SJ2Q 10494 EC50 >= 18900 nM T88505 D0X4IO 5350 EC50 = 580 nM T86717 CI0WH9 72 Ki = 44000 nM T86717 CQSM62 2556 Ki = 5.4 nM T86717 CC0GY6 10106750 Ki = 1700 nM T86717 CP24TU 10354627 Ki = 350 nM T86717 CW5MS1 11820665 Ki = 90000 nM T86717 C97THC 44277278 Ki = 220 nM T86717 C69LJX 44277306 Ki = 540 nM T86717 C85NKC 44387186 Ki = 220 nM T86717 D07QJJ 289 Ki = 630000 nM T49072 D0PQ8T 9846574 IC50 = 158.49 nM T49072 D08FGX 10173280 IC50 < 5 nM T49072 C63COK 9907171 EC50 = 251.19 nM T49072 C16EGD 10119115 Ki = 41 nM T49072 C27NVQ 10119117 IC50 = 134 nM T49072 CIM39E 10121972 Ki = 3 nM T49072 CV38OW 10123931 EC50 = 1.8 nM T49072 COJ2T3 10190075 Ki = 12 nM T49072 CJ0A6T 10210584 Ki = 140 nM T49072 CZU31E 10213684 EC50 = 3 nM T49072 C9RE3X 10230399 Ki = 158.49 nM T49072 CSZN34 10232516 Ki = 71 nM T49072 CG2NX0 10303115 IC50 = 67 nM T49072 C9Y0VH 10407901 EC50 = 1148.15 nM T49072 CRI6W5 10474282 EC50 = 4000 nM T49072 CV9N3J 10931175 Ki = 0.1995 nM T49072 CCKN40 11272107 IC50 = 23 nM T49072 C1MW2B 11318295 IC50 = 3.6 nM T49072 CBM63Z 11325792 EC50 = 134.9 nM T49072 C6L3BU 11480204 Ki = 1995.26 nM T49072 CFU13E 11495815 EC50 = 2137.96 nM T49072 C80CTR 11496131 EC50 = 4265.8 nM T49072 C9HO4S 11496252 EC50 = 6456.54 nM T49072 C9U3SA 11501947 EC50 = 275.42 nM T49072 C23AVP 11508921 EC50 = 1698.24 nM T49072 C3VZF6 11510666 EC50 = 1778.28 nM T49072 C1IZ9U 11520939 Ki = 5.012 nM T49072 C4QR1M 11524599 EC50 = 1862.09 nM T49072 CD43QM 11524788 EC50 = 524.81 nM T49072 CA4JN5 11525327 EC50 = 5128.61 nM T49072 C5MD1B 11526048 EC50 = 251.19 nM T49072 C1X6RH 11531958 EC50 = 190.55 nM T49072 CWZ53E 11532525 EC50 = 1995.26 nM T49072 COMV48 11537255 EC50 = 3548.13 nM T49072 C9IK2D 11546571 EC50 = 1548.82 nM T49072 CKAO10 11546868 EC50 = 1348.96 nM T49072 C4OL2D 11552098 EC50 = 1412.54 nM T49072 CIZ38G 11559558 EC50 = 2137.96 nM T49072 C8VRS4 11559579 EC50 = 1348.96 nM T49072 C4M8DF 11566781 EC50 = 1737.8 nM T49072 CN3T6V 11567714 EC50 = 66.07 nM T49072 CA71XO 11569119 EC50 = 1737.8 nM T49072 CJUP64 11573773 EC50 = 1995.26 nM T49072 C4VA1O 11582902 EC50 = 3630.78 nM T49072 C26HKC 11589093 EC50 = 77.62 nM T49072 C7SXO2 11591072 EC50 = 1819.7 nM T49072 C3R7KT 11595438 EC50 = 2187.76 nM T49072 C4T2UB 11604535 EC50 = 3890.45 nM T49072 CFRB75 11609885 EC50 = 2884.03 nM T49072 CQ09KY 11625650 EC50 = 144.54 nM T49072 CMG2V7 11626617 EC50 = 1122.02 nM T49072 C8Q9EN 11627432 EC50 = 269.15 nM T49072 CO2YA1 11631605 EC50 = 1348.96 nM T49072 C5U8TK 11640431 EC50 = 109.65 nM T49072 C8L4AR 11648503 EC50 = 288.4 nM T49072 CLB1S0 11653844 EC50 = 524.81 nM T49072 CIO92G 11674961 EC50 = 1659.59 nM T49072 CLH9B3 11681737 EC50 = 2290.87 nM T49072 C91ZUS 11684574 EC50 = 117.49 nM T49072 CMH71P 11696838 EC50 = 32.36 nM T49072 CO8IV2 11697064 EC50 = 2089.3 nM T49072 CQ42XD 11829173 Ki = 0.2512 nM T49072 CL7U4R 11983241 EC50 = 128.82 nM T49072 CN2C7Y 11993926 Ki = 2.951 nM T49072 C1MUC6 11993927 Ki = 0.912 nM T49072 CG8M6Q 11994050 Ki = 10 nM T49072 CS2ZL4 11994174 Ki = 407.38 nM T49072 CD1W6E 11994175 Ki < 10000 nM T49072 C9RI2A 11994176 Ki = 19.5 nM T49072 CJW87H 11995279 Ki = 2.239 nM T49072 CXUB81 11995367 Ki = 1.622 nM T49072 CYW3N8 11995368 Ki = 74.13 nM T49072 CNV8G4 11995466 Ki = 9.12 nM T49072 C7ECR0 11995574 Ki = 131.83 nM T49072 CU8VD4 11995576 Ki = 154.88 nM T49072 CB58NF 12052408 Ki = 501.19 nM T49072 C7V3GE 12052410 Ki = 501.19 nM T49072 CEAV96 12052411 Ki = 501.19 nM T49072 C5Q6DK 12052412 Ki = 630.96 nM T49072 C5CML8 12052413 Ki = 794.33 nM T49072 CVZ8E4 12052415 Ki = 630.96 nM T49072 CO57KE 12052419 Ki = 199.53 nM T49072 C9W2YP 12704866 Ki = 12.59 nM T49072 CAZ2K4 12704868 Ki > 7943.28 nM T49072 C64RPT 15959612 Ki = 2.399 nM T49072 C2BO1Y 15983196 EC50 = 1288.25 nM T49072 CHUJ96 15983198 EC50 = 2754.23 nM T49072 C1KU5G 15983200 EC50 = 1148.15 nM T49072 C70NQD 15983311 EC50 = 1949.84 nM T49072 C4T5PJ 15983313 EC50 = 1122.02 nM T49072 CQ4B3L 15983315 EC50 = 1071.52 nM T49072 C8LV3Z 15983317 EC50 = 1862.09 nM T49072 C64NLP 15983319 EC50 = 467.74 nM T49072 C74QSP 15983321 EC50 = 2511.89 nM T49072 C7PQH6 15983323 EC50 = 2290.87 nM T49072 CP15MN 15983325 EC50 = 1380.38 nM T49072 CPA25I 15983441 EC50 = 870.96 nM T49072 C2S6UO 15983443 EC50 = 1513.56 nM T49072 C4Q8DN 15983445 EC50 = 1659.59 nM T49072 CO94FQ 15983447 EC50 = 1122.02 nM T49072 C3QD7J 15983449 EC50 = 2951.21 nM T49072 CTE1B0 15983558 EC50 = 512.86 nM T49072 C5V7YR 15983560 EC50 = 398.11 nM T49072 C10UQP 15983562 EC50 = 4168.69 nM T49072 CN3RZ7 15983564 EC50 = 1122.02 nM T49072 CX90QS 15983566 EC50 = 5888.44 nM T49072 C2ZL6V 15983568 EC50 = 4570.88 nM T49072 CBZ9U8 15983570 EC50 = 2290.87 nM T49072 CSM32N 15983684 EC50 = 5370.32 nM T49072 CP81BL 15983686 EC50 = 1548.82 nM T49072 CT8DN3 15983688 EC50 = 436.52 nM T49072 C03FAM 15983690 EC50 = 1995.26 nM T49072 CY7EU5 15983691 EC50 = 3090.3 nM T49072 CO7DB5 15983693 EC50 = 1737.8 nM T49072 C2BY5A 15983695 EC50 = 575.44 nM T49072 C9E2QK 15983816 EC50 = 602.56 nM T49072 CAM1D2 15983818 EC50 = 371.54 nM T49072 CV45UJ 15983820 EC50 = 1412.54 nM T49072 CVOM82 15983822 EC50 = 134.9 nM T49072 CFHL19 15983824 EC50 = 588.84 nM T49072 C36FMO 15983826 EC50 = 380.19 nM T49072 C6QFA3 16126405 EC50 = 426.58 nM T49072 C6XI8K 16126557 EC50 = 457.09 nM T49072 CBHE06 16656749 Ki = 45 nM T49072 CCI3R4 18613636 Ki = 500 nM T49072 COL28T 23627249 Ki = 76 nM T49072 CYAI24 23627251 Ki = 3200 nM T49072 CU37SO 23627305 Ki = 200 nM T49072 C59IEM 23627492 Ki = 310 nM T49072 CIC1B2 23627554 Ki = 160 nM T49072 CS47WY 23627555 Ki = 230 nM T49072 CTK04S 23627556 Ki = 160 nM T49072 CHP24B 23627557 Ki = 310 nM T49072 C38DAG 23627613 Ki = 310 nM T49072 C0Y3TV 23627666 Ki = 13 nM T49072 C32ODJ 23627722 Ki = 49 nM T49072 CH3B6T 23728637 Ki = 65 nM T49072 CZG49M 24795079 EC50 = 22.91 nM T49072 C39CUI 24804161 Ki = 77 nM T49072 CMR3S5 24804323 Ki = 30 nM T49072 C1ZPK6 24804324 Ki = 27 nM T49072 CT90MW 24804325 Ki = 160 nM T49072 C93BWM 24804326 Ki = 54 nM T49072 CAG98B 24804491 Ki = 140 nM T49072 CP9RX7 24804816 Ki = 430 nM T49072 CM80JI 24863522 Ki = 4 nM T49072 CI53SE 24893978 IC50 = 4 nM T49072 CS9IJ7 24952349 EC50 = 575.44 nM T49072 CSPJ97 24952350 EC50 = 436.52 nM T49072 C7K8XM 24952351 EC50 = 575.44 nM T49072 CZWN41 24952352 EC50 = 363.08 nM T49072 C0X6CK 24952353 EC50 = 75.86 nM T49072 CXK90H 24952706 EC50 = 74.13 nM T49072 CICR58 24952707 EC50 = 309.03 nM T49072 CIU2V1 24952708 EC50 = 812.83 nM T49072 CWJS29 24952709 EC50 = 645.65 nM T49072 CQX43B 24952710 EC50 = 1071.52 nM T49072 CXU41F 24953055 EC50 = 125.89 nM T49072 C9L2QI 24953056 EC50 = 346.74 nM T49072 CH5K1N 24953057 EC50 = 812.83 nM T49072 CXW59P 24953058 EC50 = 537.03 nM T49072 CYI4J0 24953059 EC50 = 1096.48 nM T49072 C8TIJ2 24953060 EC50 = 3467.37 nM T49072 CNX02I 24953410 EC50 = 43.65 nM T49072 C6OKC2 24953411 EC50 = 104.71 nM T49072 COG8F1 24953412 EC50 = 524.81 nM T49072 CM67NG 24953413 EC50 = 6456.54 nM T49072 CEBS42 24953414 EC50 = 3801.89 nM T49072 CGA1L2 24954830 EC50 = 199.53 nM T49072 CH9P0Y 24954831 EC50 = 120.23 nM T49072 CHR4O0 24955187 EC50 = 870.96 nM T49072 CD21XO 24955189 EC50 = 741.31 nM T49072 C10OTZ 24955192 EC50 = 2754.23 nM T49072 CHWQ64 25067045 Ki = 3.981 nM T49072 CA76KJ 25067046 Ki = 6 nM T49072 C7YRG0 25067560 Ki = 3.981 nM T49072 CT85IU 25124736 Ki = 11 nM T49072 CD26MZ 25125075 Ki < 5 nM T49072 CHWF98 25125422 Ki = 4 nM T49072 CS46EK 25125764 Ki = 18 nM T49072 CP83IT 25126424 Ki = 18 nM T49072 C8XY4N 25126427 Ki = 4 nM T49072 C49ESA 25127070 Ki = 59 nM T49072 CS7P2F 25127071 Ki = 11 nM T49072 CP53WS 25127072 Ki = 44 nM T49072 CL38JC 25128051 Ki < 6 nM T49072 C9VQ1W 25211348 Ki = 63.1 nM T49072 CLG9B0 44206680 Ki = 64 nM T49072 C9X7MD 44290317 Ki = 0.7943 nM T49072 CJIH40 44296160 EC50 = 3.6 nM T49072 C6TY7M 44296161 EC50 = 2.4 nM T49072 CV45HJ 44296244 EC50 = 2.3 nM T49072 CF1MP6 44296245 EC50 = 2.5 nM T49072 C0B7GR 44296304 EC50 > 10000 nM T49072 CNQY76 44296305 EC50 = 3.8 nM T49072 C8RE9A 44296314 EC50 = 1.8 nM T49072 C4HW2X 44296318 EC50 = 1003 nM T49072 C62BNG 44296607 EC50 > 10000 nM T49072 CVS92U 44296608 EC50 = 53 nM T49072 C92KCB 44399055 Ki < 10000 nM T49072 C7I2TY 44399056 Ki < 10000 nM T49072 CG5HJ8 44399057 Ki < 10000 nM T49072 C1QYR9 44399062 Ki = 398.11 nM T49072 CM6RZ4 44399063 Ki = 125.89 nM T49072 COUH52 44399075 Ki < 10000 nM T49072 CSK83U 44399082 Ki < 10000 nM T49072 CQ27YD 44399083 Ki = 2511.89 nM T49072 C56XIU 44399084 Ki = 398.11 nM T49072 CO60UE 44399085 Ki < 10000 nM T49072 CK7P3O 44399093 Ki = 398.11 nM T49072 CF2T0Q 44399094 Ki = 630.96 nM T49072 C4YKS5 44399136 Ki < 10000 nM T49072 CJ14UC 44399152 Ki < 10000 nM T49072 CUHC02 44399163 Ki = 316.23 nM T49072 CP83MT 44399166 Ki = 1995.26 nM T49072 CRN95C 44399167 Ki < 10000 nM T49072 C07RXT 44399168 Ki = 251.19 nM T49072 CUA85N 44399169 Ki = 2511.89 nM T49072 C7FV5M 44399216 Ki < 10000 nM T49072 C3FG6O 44399217 Ki < 10000 nM T49072 C7PUT2 44399234 Ki = 2511.89 nM T49072 C3Y0VF 44399243 Ki < 10000 nM T49072 CA78BQ 44399254 Ki = 1000 nM T49072 C4XYI8 44399255 Ki < 10000 nM T49072 CI7C4B 44399268 Ki < 10000 nM T49072 CSEL71 44399271 Ki < 10000 nM T49072 CMW5O6 44399398 Ki = 630.96 nM T49072 CCB5T6 44399453 Ki = 3162.28 nM T49072 CZ7AL0 44399475 Ki = 1995.26 nM T49072 C6YZ9B 44399476 Ki = 2511.89 nM T49072 C57UZK 44400855 EC50 = 6300 nM T49072 C9Z1HC 44409467 EC50 = 1445.44 nM T49072 CT7LZ1 44409477 EC50 = 407.38 nM T49072 CR9K0Z 44409478 EC50 = 1023.29 nM T49072 C8OD5I 44409534 EC50 = 1513.56 nM T49072 CW09SJ 44409548 EC50 = 5011.87 nM T49072 CM78VG 44417524 Ki = 2.884 nM T49072 C57VIK 44417525 Ki = 1.122 nM T49072 C2RT1P 44417526 Ki = 23.44 nM T49072 C3AIY4 44417527 Ki < 10000 nM T49072 CQD80R 44421620 Ki = 0.2512 nM T49072 C2S3HW 44421621 Ki = 0.1995 nM T49072 CDJ3Z5 44421622 Ki = 1.259 nM T49072 CJ8ES1 44421623 Ki = 1.259 nM T49072 CP0EQ1 44421624 Ki = 15.85 nM T49072 CM5JF8 44421625 Ki = 10 nM T49072 CLD6O0 44421626 Ki = 12.59 nM T49072 CBKQ13 44421627 Ki = 398.11 nM T49072 CV69SU 44435044 Ki = 30 nM T49072 C0S6QL 44448289 Ki = 794.33 nM T49072 CJR95K 44448290 Ki = 100 nM T49072 CD18IM 44448293 Ki = 501.19 nM T49072 CXZ4F5 44448314 Ki = 158.49 nM T49072 CT39GZ 44448315 Ki = 79.43 nM T49072 C7EQ5Z 44448316 Ki = 79.43 nM T49072 C5D7TB 44448317 Ki = 199.53 nM T49072 C1J6NP 44448337 Ki = 1584.89 nM T49072 C15XDA 44448338 Ki = 31.62 nM T49072 CBL70O 44448339 Ki = 50.12 nM T49072 C2CBA6 44448359 Ki = 63.1 nM T49072 C8J0EO 44448361 Ki = 3162.28 nM T49072 CXFD75 44448390 Ki < 7943.28 nM T49072 C8QNY4 44448393 Ki < 7943.28 nM T49072 CCV5H2 44448394 Ki = 2511.89 nM T49072 CQ1NL8 44448396 Ki = 7943.28 nM T49072 CO8A3X 44448428 Ki = 630.96 nM T49072 CK3LV5 44448429 Ki = 79.43 nM T49072 C3SY0L 44448431 Ki = 251.19 nM T49072 CEV8L7 44448469 Ki = 15.85 nM T49072 CM0AD4 44448471 Ki = 31.62 nM T49072 C6TW2M 44448472 Ki = 7.943 nM T49072 C0U1PI 44448474 Ki = 199.53 nM T49072 CUBL60 44448510 Ki = 25.12 nM T49072 C9XA8P 44448513 Ki = 31.62 nM T49072 C4NK3Y 44448514 Ki = 199.53 nM T49072 C57UJB 44448549 Ki = 1995.26 nM T49072 CXG1Y5 44448585 Ki < 7943.28 nM T49072 C7DV3J 44448586 Ki = 794.33 nM T49072 CL1TO6 44448622 Ki < 7943.28 nM T49072 C4IJG2 44448625 Ki < 7943.28 nM T49072 CM36NZ 44448653 Ki = 1258.93 nM T49072 CR0W7C 44448656 Ki = 501.19 nM T49072 CAS5F6 44448657 Ki = 7943.28 nM T49072 CT16AC 44448691 Ki = 1584.89 nM T49072 C1G9ZO 44448692 Ki = 398.11 nM T49072 CZH84P 44448714 Ki = 1000 nM T49072 CFH7Q2 44448732 Ki = 3981.07 nM T49072 C0LBQ9 44448733 Ki = 794.33 nM T49072 CW9N0L 44448734 Ki = 3162.28 nM T49072 C50VFY 44448736 Ki = 398.11 nM T49072 CY8RO4 44448772 Ki = 79 nM T49072 C9K8EN 44448775 Ki = 16 nM T49072 CW7BG9 44448874 Ki = 6 nM T49072 CR6TO5 44448876 Ki = 1.2 nM T49072 CF40AD 44448913 Ki = 40 nM T49072 C5OR0Q 44448947 Ki = 5 nM T49072 C15VTJ 44448976 Ki = 5 nM T49072 C1F2MP 44449004 Ki = 1 nM T49072 CL9M2D 44449052 Ki = 3 nM T49072 CL4H8Y 44449053 Ki = 0.6 nM T49072 C3L4XD 44449079 Ki = 0.4 nM T49072 C4T1MQ 44449106 Ki = 0.4 nM T49072 C9XZY1 44449107 Ki = 2 nM T49072 CV31WQ 44449136 Ki = 130 nM T49072 CA4DS0 44449171 Ki = 8 nM T49072 CA61WE 44449202 Ki = 6 nM T49072 CC19LO 44449228 Ki = 2 nM T49072 C8WZ4X 44534490 Ki = 47 nM T49072 CXA81C 44534500 Ki = 108 nM T49072 CAE25R 44534504 Ki = 61 nM T49072 C1J4CS 44534506 Ki = 1500 nM T49072 C4SIT9 44534510 Ki = 230 nM T49072 C0YWB2 44534536 Ki > 10000 nM T49072 C5YR6N 44552474 EC50 = 6.94 nM T49072 C32AGV 44561123 Ki = 15 nM T49072 CONA75 44561156 Ki = 2500 nM T49072 CG1W8A 44561157 Ki = 20 nM T49072 CXH86I 44561195 Ki = 630 nM T49072 CD7A4H 44561196 Ki = 13 nM T49072 C8HCR6 44561197 Ki = 16 nM T49072 C9HG8L 44561236 Ki = 630 nM T49072 CR5T0L 44561237 Ki = 6 nM T49072 CF21JK 44561238 Ki = 3 nM T49072 CMJ60R 44561239 Ki = 0.3 nM T49072 C0W4HQ 44561240 Ki = 3 nM T49072 C6A0TH 44561276 Ki = 5 nM T49072 C23UIM 44568194 Ki > 10000 nM T49072 CA35SF 44568195 Ki > 10000 nM T49072 C74PYF 44568226 Ki = 350 nM T49072 CMK39X 44568308 Ki > 3000 nM T49072 C37SLA 44568309 Ki = 97 nM T49072 C7MN1C 44568339 Ki = 1000 nM T49072 CUZ1D9 44568368 Ki = 3500 nM T49072 CSWE21 44568369 Ki = 5.5 nM T49072 CF1EI5 44568370 Ki = 44 nM T49072 CZM49I 44568398 Ki = 10 nM T49072 C8RA4Z 44568399 Ki = 15 nM T49072 CL7WO3 44568400 Ki = 62 nM T49072 CQT5B1 44568426 Ki = 36 nM T49072 C0DM7F 44568427 Ki = 69 nM T49072 CKEA75 44568428 Ki = 42 nM T49072 CHP1V2 44568429 Ki = 120 nM T49072 CA30UC 44568484 Ki = 380 nM T49072 CQLO58 44568526 Ki = 18 nM T49072 C56PGR 44574144 Ki = 0.7943 nM T49072 CGA0R6 44574145 Ki = 1.66 nM T49072 C0BL9V 44574146 Ki = 0.2818 nM T49072 CCX54G 44574147 Ki = 19.5 nM T49072 C90IRQ 44574148 Ki = 0.8913 nM T49072 C0JCT9 44574149 Ki = 9.55 nM T49072 C78PVD 44574150 Ki = 26.3 nM T49072 C7LV2D 44574151 Ki = 3.89 nM T49072 CFR83M 44574152 Ki = 6.457 nM T49072 CA3VS1 44574153 Ki = 11.75 nM T49072 CD03JO 44574154 Ki = 13.49 nM T49072 CN4C8P 44574155 Ki = 15.85 nM T49072 CK3V7L 44574156 Ki = 2.63 nM T49072 CG2Q3J 44574157 Ki = 9.333 nM T49072 C71EGT 44574158 Ki = 9.333 nM T49072 C6YM1S 44574159 Ki = 218.78 nM T49072 CW5N9J 44580436 Ki = 1584.89 nM T49072 C9SNK2 44580437 Ki = 25.12 nM T49072 CAKQ68 44580472 Ki = 3.981 nM T49072 C67HIR 44580473 Ki = 6.31 nM T49072 CFE7C3 44580474 Ki = 794.33 nM T49072 CWCF79 44580475 Ki = 10 nM T49072 C7Q1PB 44580476 Ki = 12.59 nM T49072 CH04NR 44580477 Ki = 2511.89 nM T49072 C5NOJ6 44580515 Ki = 6.31 nM T49072 CKLS30 44580516 Ki > 7943.28 nM T49072 C92VNI 44580517 Ki = 10 nM T49072 CTXU03 44580518 Ki = 100 nM T49072 CG0W9P 44580519 Ki = 25.12 nM T49072 C7ROM9 44580563 Ki = 19.95 nM T49072 CQFS78 44580564 Ki = 12.59 nM T49072 CT8PZ9 44580565 Ki = 79.43 nM T49072 CJH8E7 44580566 Ki > 7943.28 nM T49072 CS5PQ6 44580567 Ki > 7943.28 nM T49072 C94WDR 44580568 Ki > 7943.28 nM T49072 CY4BR1 44580569 Ki > 7943.28 nM T49072 C8W0YN 44580629 Ki > 7943.28 nM T49072 C24ZOX 44580630 Ki = 794.33 nM T49072 C3N6YD 44580631 Ki = 50.12 nM T49072 CYN69E 44580632 Ki = 3981.07 nM T49072 CCU2I0 44580633 Ki = 79.43 nM T49072 CBQR53 44580634 Ki = 316.23 nM T49072 CK42PT 44580679 Ki = 100 nM T49072 CAY8O4 44580680 Ki = 794.33 nM T49072 CUK32R 44580681 Ki = 63.1 nM T49072 CFJ4O8 44580682 Ki = 50.12 nM T49072 C7UZW8 44580683 Ki = 31.62 nM T49072 CAE64R 44593421 Ki = 13 nM T49072 C85JXW 44596867 Ki = 270 nM T49072 CO3PJ1 44596869 Ki = 150 nM T49072 CBK0H3 44596870 Ki = 59 nM T49072 C68ACZ 44596964 Ki = 35 nM T49072 CCYP24 44596965 Ki = 32 nM T49072 C0KV1H 44596966 Ki = 130 nM T49072 CVNI23 44596967 IC50 = 37 nM T49072 C6SQK3 44597068 Ki = 16 nM T49072 C9XMV3 44597069 Ki = 97 nM T49072 CHA0Y7 44597070 Ki = 49 nM T49072 CL70MK 44597071 Ki = 15 nM T49072 C32OHX 44597398 Ki = 120 nM T49072 C5HME9 45481583 EC50 = 660.69 nM T49072 CV9K7O 45481596 EC50 = 316.23 nM T49072 C0GO7I 45481598 EC50 = 457.09 nM T49072 CZ14BJ 45482441 EC50 = 645.65 nM T49072 C7VR5W 45486908 Ki = 700 nM T49072 CS7G3D 45486909 Ki = 430 nM T49072 C8ITB3 45486910 Ki = 290 nM T49072 C01EUL 45486911 Ki = 540 nM T49072 CKA23P 45486916 Ki > 10000 nM T49072 CLM1Z8 45486917 Ki = 1400 nM T49072 C5LFZ3 45487731 Ki = 25 nM T49072 CO2T5A 45487747 Ki = 62 nM T49072 CAEX43 45487748 Ki = 8 nM T49072 C3G8FT 46225600 Ki = 0.7943 nM T49072 CQX8W7 46225601 EC50 = 8.51 nM T49072 CWVJ78 46225602 EC50 = 12.58 nM T49072 C0F3BR 46225603 EC50 = 13.2 nM T49072 CT7D1K 46225604 EC50 = 10.07 nM T49072 C7QXH3 46225605 EC50 = 75.66 nM T49072 C87NHE 46225606 EC50 = 20.55 nM T49072 CK5FN9 46225607 EC50 = 16.72 nM T49072 CMB78E 46897993 EC50 = 501.19 nM T49072 C83ENG 46897994 EC50 = 691.83 nM T49072 C2QOX3 46897995 EC50 = 263.03 nM T49072 C0QPO8 46897996 EC50 = 2290.87 nM T49072 C6PUL2 46897997 EC50 = 1174.9 nM T49072 CEQ1Z4 46897998 EC50 = 2238.72 nM T49072 C0U1BK 46897999 EC50 = 51.29 nM T49072 CO58CR 46907359 Ki = 12 nM T49072 CJVI15 49798794 EC50 = 4168.69 nM T49072 C5BA4U 49798987 EC50 = 1737.8 nM T49072 CH14NE 49798989 EC50 = 933.25 nM T49072 CG0O7K 49799023 EC50 = 724.44 nM T49072 C2IH4V 49799029 EC50 = 1412.54 nM T49072 CO9PH7 49799137 EC50 = 954.99 nM T49072 C8BCG3 49799280 EC50 = 1949.84 nM T49072 CZ6Q3U 49799289 EC50 = 147.91 nM T49072 C4XLI7 49799291 EC50 = 2884.03 nM T49072 CG5RU6 49799325 EC50 = 1148.15 nM T49072 CP2NQ0 49799327 EC50 = 2398.83 nM T49072 C4WDH8 49799329 EC50 = 5248.07 nM T49072 CR2J4L 49799366 EC50 = 676.08 nM T49072 CO34HB 49799368 EC50 = 2951.21 nM T49072 CC50RX 49799485 EC50 = 3801.89 nM T49072 C1H4EZ 71579743 IC50 = 34 nM T49072 C46EMS 71579744 IC50 = 742 nM T49072 CKE13T 71579745 IC50 = 245 nM T49072 C74HVJ 71579746 IC50 = 440 nM T49072 CL4XV9 71579747 IC50 = 237 nM T49072 CVS52I 71579748 IC50 = 1450 nM T49072 CZ2EP0 71579838 IC50 = 669 nM T49072 CAC61T 71579839 IC50 = 3060 nM T49072 C6QOY1 71579840 IC50 = 1300 nM T49072 CNR2B7 71579842 IC50 > 10000 nM T49072 CE9MZ2 71579843 IC50 = 3500 nM T49072 C9T2XZ 71579935 IC50 = 765 nM T49072 CN0QH7 71580033 IC50 > 5000 nM T49072 C1YL0G 71580034 IC50 = 120 nM T49072 CDBE78 71580035 IC50 = 6200 nM T49072 CHFR07 71580133 IC50 = 840 nM T49072 C2B0KV 71580134 IC50 = 350 nM T49072 CI5RP8 71580135 IC50 = 2100 nM T49072 C4LAH1 71580136 IC50 > 10000 nM T49072 CU9ES1 71716535 IC50 = 620 nM T49072 CR6A8G 71717139 IC50 = 1870 nM T49072 C7V2EJ 71717140 IC50 = 1130 nM T49072 C41CPY 71718372 IC50 = 714 nM T49072 CW9N3H 71718978 IC50 = 550 nM T49072 CD26WI 71719581 IC50 = 191 nM T49072 CTGR27 71719582 IC50 = 180 nM T49072 CP8D7M 71720174 IC50 = 950 nM T49072 CXA76T 71720175 IC50 = 2000 nM T49072 C3W5ZV 72792556 IC50 = 361 nM T49072 C4CX1G 72792624 IC50 = 29 nM T49072 CTJ7L1 72792625 IC50 = 27.54 nM T49072 CI5L8P 72792626 IC50 = 10 nM T49072 CZD74C 72792689 IC50 = 21 nM T49072 CMC19D 72792690 IC50 > 0.00001 nM T49072 CW5P8C 72792691 IC50 = 89.13 nM T49072 C3Q8OK 72792760 IC50 > 0.00001 nM T49072 CUHN72 72793454 EC50 = 2.692 nM T49072 C1LUB7 72793455 IC50 = 16.98 nM T49072 C2W7XO 72793456 IC50 = 46 nM T49072 CQPH62 72793526 IC50 = 58 nM T49072 C1TR0M 72793527 IC50 = 181 nM T49072 CNV3X9 72793528 IC50 > 0.00001 nM T49072 CBM23K 72793598 IC50 > 0.000001 nM T49072 C5X8VR 72793599 IC50 = 281.84 nM T49072 CL9WO8 72793600 IC50 = 8.913 nM T49072 CZ7H2U 73345733 EC50 = 1.9 nM T49072 CVE47Z 73350122 Ki = 12.59 nM T49072 C0IQD5 73350313 EC50 = 14800 nM T49072 C2K8UI 73351822 EC50 = 193 nM T49072 CAR20D 73351823 EC50 = 1303 nM T49072 CO0TN2 73353299 EC50 = 233 nM T49072 C82UXW 73353300 EC50 = 2.7 nM T49072 COS0J7 73354813 EC50 = 3.3 nM T49072 CUSI09 73354814 EC50 = 3.2 nM T49072 CS83ZT 73356165 Ki = 1.259 nM T49072 C9ODC3 73356323 Ki = 12.59 nM T49072 CR0N4T 73356357 EC50 = 1.8 nM T49072 CA47SW 73356358 EC50 = 5.7 nM T49072 CIA5Q7 76310152 IC50 = 808 nM T49072 CMQ92X 76321099 IC50 = 60 nM T49072 C0I8DT 76331986 IC50 > 0.00001 nM T49072 C2D7GV 86291694 IC50 = 3220 nM T49072 C4Q0YD 86291695 IC50 = 1230 nM T49072 CIRF10 86291696 IC50 = 26 nM T49072 C78VQK 86291697 IC50 = 60 nM T49072 CD8OY0 86291904 IC50 = 20 nM T49072 CJ9HZ1 86291905 IC50 = 42 nM T49072 CHF06S 86291906 IC50 = 20 nM T49072 CI47WB 86291907 IC50 = 140 nM T49072 CTRA15 86291908 IC50 = 190 nM T49072 CO74AR 86292101 IC50 = 13 nM T49072 C17OVD 86292104 IC50 = 36 nM T49072 CVX6I0 86294592 IC50 = 78 nM T49072 CGBL14 86305736 IC50 = 160 nM T49072 CQSO57 86305831 IC50 = 600 nM T49072 C6GLM8 118708005 Ki = 1.995 nM T49072 CJFR71 118708006 Ki = 0.7244 nM T49072 C1TD5M 118708007 Ki = 0.3981 nM T49072 C0CGL3 118708008 Ki = 6.457 nM T49072 CS6UT8 118708009 Ki = 1.738 nM T49072 CZJE89 118708010 Ki = 12.88 nM T49072 CA5FW7 118708011 Ki = 1.23 nM T49072 CM2H8C 118708012 Ki = 1.047 nM T49072 C2U8WF 118708013 Ki = 0.7762 nM T49072 C93MZQ 118708014 Ki = 2.239 nM T49072 CJY61S 118708015 Ki = 1.82 nM T49072 CCT3Y2 118708016 Ki = 12.02 nM T49072 C5DNX0 118708017 Ki = 1.778 nM T49072 CVGL96 118708018 Ki = 16.98 nM T49072 CYIB53 118723009 IC50 = 220 nM T49072 CT21PB 118723010 IC50 = 2140 nM T49072 CK2OJ1 118723011 IC50 = 450 nM T49072 C8QEN1 118723012 IC50 = 930 nM T49072 CXW4K0 123185525 IC50 = 140 nM T49072 C18EXT 123264706 IC50 = 80 nM T49072 CBV79A 123794584 IC50 = 49 nM T49072 C9EBM4 123922871 IC50 = 74 nM T49072 C7J6VZ 127048901 IC50 > 1000 nM T49072 C2RJ5G 127049894 IC50 > 1000 nM T49072 CDZ4G1 127050201 IC50 > 1000 nM T49072 C92OKY 127051389 IC50 > 1000 nM T49072 CA72KD 127051713 IC50 > 1000 nM T49072 CT5P9H 127052350 IC50 > 1000 nM T49072 CZG26S 134133034 IC50 = 140 nM T49072 CW6MA1 134133573 IC50 = 51 nM T49072 CPJ9L6 134134886 IC50 = 100 nM T49072 CJ1P9I 134138102 IC50 = 970 nM T49072 C4CP1I 134140417 IC50 = 610 nM T49072 CWA53M 134141359 IC50 = 53 nM T49072 C3R6QC 134141963 IC50 = 63 nM T49072 CRS17M 134142270 IC50 = 560 nM T49072 CV73EA 134142581 IC50 = 86 nM T49072 C7IJQ4 134146007 IC50 = 770 nM T49072 C7OX1A 134148271 IC50 = 310 nM T49072 CP5OJ9 134151328 IC50 = 74 nM T49072 C5LGF1 134151441 IC50 = 90 nM T49072 CQ34TM 134151496 IC50 = 25 nM T49072 CB4ES7 134152171 IC50 = 49 nM T49072 CVH8A7 134152840 IC50 = 130 nM T49072 CF9LO8 134153111 IC50 = 340 nM T49072 C7GDL0 134155324 IC50 = 100 nM T49072 CA9MB3 134156076 IC50 = 120 nM T49072 CNE10K 134156326 IC50 = 180 nM T49072 CRYM82 134156353 IC50 = 87 nM T49072 C8M5ZD 135747623 Ki = 1.738 nM T49072 CRQF20 135747625 Ki > 10000 nM T49072 C8QG3A 137631910 EC50 = 5.012 nM T49072 COR5B1 137638373 EC50 = 7.079 nM T49072 CYF3V9 137649718 EC50 = 6.166 nM T49072 CTY73A 137659347 EC50 = 4.169 nM T49072 C70YKO 142747238 IC50 = 33 nM T49072 C0N9OB 142747242 IC50 = 80 nM T49072 CCX47N 142747243 IC50 = 120 nM T49072 C96GUQ 142747247 IC50 = 20 nM T49072 CH12MA 142747251 IC50 = 61 nM T49072 C1WHG7 142747252 IC50 = 24 nM T49072 CT5ZS4 142747253 IC50 = 34 nM T49072 CGP6I3 142747254 IC50 = 24 nM T49072 C6C5YL 142747255 IC50 = 14 nM T49072 CP2KV1 142747256 IC50 = 15 nM T49072 CAJG01 142747258 IC50 = 68 nM T49072 CJB48D 142747265 IC50 = 120 nM T49072 CPU93E 142747268 IC50 = 60 nM T49072 C8K4YZ 142747271 IC50 = 80 nM T49072 C1Q7LB 142747273 IC50 = 330 nM T49072 CYM6E9 142747275 IC50 = 15 nM T49072 C0IF5W 142747279 IC50 = 31 nM T49072 CU2ZG4 142747281 IC50 = 15 nM T49072 CN5R6Z 142747285 IC50 = 18 nM T49072 CZW83T 142747289 IC50 = 48 nM T49072 CD9MV0 142747291 IC50 = 26 nM T49072 C3MI8P 142747294 IC50 = 6 nM T49072 C76UOQ 142747296 IC50 = 15 nM T49072 CUWI61 142747298 IC50 = 66 nM T49072 C3P4UM 142747303 IC50 = 38 nM T49072 CA17CO 145965592 EC50 = 46.77 nM T49072 CX08NI 145966260 IC50 = 26.92 nM T49072 CBZ63S 145967082 EC50 = 660.69 nM T49072 CO67QF 145973104 EC50 = 10.72 nM T49072 C1GM8I 145973990 EC50 = 380.19 nM T49072 CMTJ57 145977223 EC50 = 15.14 nM T49072 C1JO7S 145977587 EC50 = 53.7 nM T49072 C8O1JF 145978068 IC50 = 3.981 nM T49072 CR3N0U 148470142 IC50 = 48 nM T49072 C58XIL 155512483 IC50 = 43 nM T49072 C1O7RM 155519842 EC50 = 104.71 nM T49072 CYUX46 155520913 Ki = 48.98 nM T49072 CAO4G6 155524087 Ki = 3.548 nM T49072 C1DGH0 155524911 Ki = 2137.96 nM T49072 C3XED8 155529504 Ki = 3.548 nM T49072 CR2A5D 155532198 EC50 = 22.39 nM T49072 C63OCP 155536007 Ki = 1.738 nM T49072 CRG03B 155537097 EC50 = 2.692 nM T49072 C7GCN0 155537736 EC50 = 5.623 nM T49072 C10NRL 155540766 Ki = 1513.56 nM T49072 CJB42E 155543279 IC50 = 9 nM T49072 C1VS8U 155544020 Ki = 2.188 nM T49072 CKG3O8 155549850 Ki > 10000 nM T49072 C89PVN 155550733 Ki = 2089.3 nM T49072 CTIQ47 155552384 IC50 = 120 nM T49072 CCJ2D9 155560178 Ki = 5370.32 nM T49072 C3IYP8 155560750 EC50 = 18.62 nM T49072 C76BQA 155567837 Ki = 2.951 nM T49072 D00CLB 10120078 Ki = 110 nM T49072 D03SAV 3082718 Ki = 4000 nM T49072 D04UHT 11995575 Ki = 263.03 nM T49072 D07JDU 21023902 Ki = 5.4 nM T49072 D0M9ZX 11663047 EC50 = 77.62 nM T49072 D0R8GW 9797568 EC50 = 250 nM T49072 D0T0RI 23627612 Ki = 570 nM T32972 D00AXJ 4189 IC50 = 200 nM T32972 D00BCP 2727 IC50 > 200000 nM T32972 D01AQT 441383 IC50 = 3000 nM T32972 D02NTO 5510 IC50 = 50000 nM T32972 D02YIZ 12560 IC50 > 200000 nM T32972 D06OIV 5505 IC50 > 200000 nM T32972 D06WTZ 53232 IC50 > 200000 nM T32972 D06XMU 6013 IC50 = 50000 nM T32972 D07BSQ 5994 IC50 > 200000 nM T32972 D09GOS 2812 IC50 = 130 nM T32972 D09LNI 3365 IC50 = 0.042 ug.mL-1 T32972 D0A2ZX 4173 IC50 > 200000 nM T32972 D0A4YE 5335 IC50 > 200000 nM T32972 D0AA2D 2378 IC50 = 342 nM T32972 D0B4RU 8955 IC50 > 200000 nM T32972 D0C1SF 441140 IC50 = 50000 nM T32972 D0EV8E 3198 IC50 = 50 nM T32972 D0G3DL 135398735 IC50 = 30000 nM T32972 D0J2KV 4932 IC50 > 200000 nM T32972 D0S4BR 1349907 IC50 > 200000 nM T32972 D03TFJ 5798 IC50 > 200000 nM T32972 CY4WG9 3793 IC50 = 0.06 ug.mL-1 T32972 C9LCD8 3823 Ki = 24.5 nM T32972 C7TQ5V 33605 IC50 > 10000 nM T32972 CWTQ15 43233 IC50 > 10000 nM T32972 C67HRU 9803497 IC50 = 800 nM T32972 CV36QP 9863489 IC50 = 0.01 ug.mL-1 T32972 CH59XL 9950501 IC50 = 0.032 ug.mL-1 T32972 CZG39B 10067630 IC50 = 0.032 ug.mL-1 T32972 C87HAM 10574415 IC50 = 3100 nM T32972 CT9D4K 15521016 IC50 > 200000 nM T32972 CZX08M 25142015 Ki = 17.7 nM T32972 C3MJC2 44297152 IC50 = 0.01 ug.mL-1 T32972 C3E8SA 44297154 IC50 = 0.032 ug.mL-1 T32972 CR41DF 44297155 IC50 = 0.049 ug.mL-1 T32972 C3NGY0 44297160 IC50 = 0.024 ug.mL-1 T32972 C3ZP5V 44297175 IC50 = 0.026 ug.mL-1 T32972 CRT72J 44297203 IC50 = 0.054 ug.mL-1 T32972 CE9P5R 44376591 IC50 = 0.08 ug.mL-1 T32972 C3MDA2 44450698 IC50 = 4500 nM T32972 C89QBR 44450722 IC50 = 2500 nM T32972 C0T3OG 44450765 IC50 > 200000 nM T32972 CN3B9F 44450766 IC50 > 200000 nM T32972 CFJ67L 44450780 IC50 = 100000 nM T32972 CM91HP 44450781 IC50 = 1300 nM T32972 CWQ27L 44450782 IC50 = 100000 nM T32972 C5RC9L 44450783 IC50 = 910 nM T32972 C1CD4Z 44450787 IC50 = 75000 nM T32972 C91MSE 44450821 IC50 = 26000 nM T32972 C5DIR3 44450822 IC50 = 9700 nM T32972 C6G9JD 119081677 IC50 < 500 nM T32972 CY5I6G 139592939 IC50 < 1000 nM T32972 C6E1CP 145984384 IC50 < 500 nM T32972 CEFJ07 155510992 IC50 < 500 nM T32972 COP1N7 155513568 IC50 < 500 nM T32972 CIP3V9 155517098 IC50 < 500 nM T32972 CXPR45 155523005 IC50 = 5200 nM T32972 CKQY16 155526985 IC50 = 1500 nM T32972 CQL2I4 155528519 IC50 < 500 nM T32972 CEZ6L5 155531616 IC50 < 500 nM T32972 C4M7FI 155535954 IC50 = 12000 nM T32972 CLF1C5 155569610 IC50 = 3000 nM T32972 D00UMG 44450788 IC50 = 300 nM T32972 D02DLW 5997 IC50 > 200000 nM T32972 D0A9PS 5281969 IC50 > 200000 nM T32972 D0HD9P 444899 IC50 > 200000 nM T32972 D0S0AN 444746 IC50 = 4000 nM T16308 D02DGU 444795 IC50 = 820 nM T16308 D0C0NH 3806 IC50 = 10120 nM T16308 D0U2BH 65064 IC50 = 20000 nM T16308 CV2U9A 65708 IC50 > 10000 nM T16308 C5KG0T 69762 Ki = 50 nM T16308 CQ2BF9 120065 IC50 = 360000 nM T16308 CT61NR 221007 IC50 = 1460 nM T16308 C24QJI 259188 IC50 = 16000 nM T16308 CFM52S 643974 IC50 = 1500 nM T16308 C0NO6B 665156 IC50 = 720000 nM T16308 CW5E8J 776315 IC50 > 1000000 nM T16308 CEI60J 1516859 IC50 = 63000 nM T16308 CO83ED 3163396 IC50 = 630000 nM T16308 C6KX2V 5172700 IC50 = 2230 nM T16308 C9F2NB 6022998 Ki = 625.2 nM T16308 CHO2E7 7147232 IC50 > 100000 nM T16308 CM27DZ 7147236 IC50 > 100000 nM T16308 CQ52DW 7147253 IC50 > 100000 nM T16308 C4XAI7 10395243 IC50 = 1000 nM T16308 CO2RJ8 11181229 IC50 = 800 nM T16308 CNLB28 11234712 Ki = 179 nM T16308 C7G8NB 11400021 IC50 = 1500 nM T16308 C4T6HL 11418384 IC50 = 6 nM T16308 CYB60N 11510199 Ki = 12 nM T16308 CKHV17 11510716 Ki = 196 nM T16308 CE8N7V 11549962 IC50 = 22000 nM T16308 C2ZN7F 11581756 Ki = 76 nM T16308 C0DQO3 11590467 Ki = 580 nM T16308 C2AE0B 11615117 Ki = 1.2 nM T16308 C8N2TD 11655448 Ki = 320 nM T16308 CK13LM 11675244 Ki = 80 nM T16308 C67ZGX 11689343 Ki = 138 nM T16308 CH5L9O 11689942 Ki = 1360 nM T16308 C4Q9RT 11718765 Ki = 75 nM T16308 CZK2J3 11749915 Ki = 32 nM T16308 CUR37N 11750082 Ki = 57 nM T16308 CH7YU6 11773558 Ki = 100 nM T16308 CDW2O9 12875050 IC50 > 100000 nM T16308 CKMU35 13154044 IC50 = 450000 nM T16308 CG7XU3 14186396 Ki = 28000 nM T16308 CI3VR1 15559100 IC50 = 13160 nM T16308 CL6FK8 16093559 Ki = 200 nM T16308 C2GN6Y 16093564 IC50 = 5600 nM T16308 CE19XA 16115228 Ki = 9000 nM T16308 CLSK31 43445097 IC50 = 23000 nM T16308 C3A2IN 44263408 Ki > 50000 nM T16308 CH1NI3 44263409 Ki = 1700 nM T16308 C6U3LF 44263410 Ki = 9460 nM T16308 CFU9J5 44263411 Ki = 8770 nM T16308 COJ6H5 44263413 Ki = 525 nM T16308 C9OUT8 44263414 Ki = 78 nM T16308 C0O3BJ 44263415 Ki = 89 nM T16308 CS3AY9 44409458 IC50 = 8000 nM T16308 CXGA65 44409459 IC50 = 25000 nM T16308 C3N2XM 44409485 IC50 = 15000 nM T16308 CPWY39 44409486 Ki = 4.8 nM T16308 CF5G0W 44409493 IC50 = 7000 nM T16308 CA70JB 44409494 IC50 = 20000 nM T16308 CCMO58 44409513 Ki = 183 nM T16308 CD4AN3 44409545 IC50 > 50000 nM T16308 C8XG3E 44409546 IC50 > 50000 nM T16308 CBP40A 44409547 IC50 = 30000 nM T16308 CMS19Z 44409586 IC50 > 50000 nM T16308 CCK72B 44409587 IC50 = 20000 nM T16308 C0D7AX 44409639 IC50 = 10000 nM T16308 CU81EC 44409640 IC50 = 15000 nM T16308 CU16CS 44444615 IC50 = 28300 nM T16308 C6V4UK 44517642 IC50 = 7500 nM T16308 COK0H9 44517643 IC50 = 830 nM T16308 CT3F0E 44517644 IC50 = 6600 nM T16308 C4FUQ2 44517646 IC50 = 3900 nM T16308 C3JPG8 45114305 Ki = 12000 nM T16308 C7TBY3 45157073 IC50 = 270000 nM T16308 CDG5O7 45379213 IC50 = 43 nM T16308 CCLH68 45379353 IC50 = 63000 nM T16308 CN2FZ9 45379355 IC50 = 220 nM T16308 C8W2AU 45379505 IC50 = 1100 nM T16308 C0LTV1 45486927 Ki = 4130 nM T16308 C8I7OD 46191373 IC50 = 25 nM T16308 C4M3XB 46191374 IC50 = 2600 nM T16308 C14SFO 46227798 IC50 = 78000 nM T16308 CAY1K0 46227799 IC50 = 320 nM T16308 C7QIN6 46227804 IC50 = 180 nM T16308 CO6YP2 46227805 IC50 = 25 nM T16308 C3F9WP 46227807 IC50 = 6300 nM T16308 C7L0JB 46227808 IC50 = 260 nM T16308 C3OMF6 46227817 IC50 = 10000 nM T16308 CAH78N 46227819 IC50 > 2000000 nM T16308 CJ6IN7 46227822 IC50 = 130 nM T16308 C4TU0L 46227823 IC50 = 92000 nM T16308 CUZS16 46883910 Ki = 6 nM T16308 CPD6Z2 46883912 Ki = 179 nM T16308 C4J1CO 46883947 Ki = 93000 nM T16308 CZV83L 46883948 Ki = 63000 nM T16308 CY39VT 46883949 Ki = 351000 nM T16308 C4NW1U 46884010 Ki = 103000 nM T16308 C0W5IK 46884011 Ki = 5700 nM T16308 C6F5DQ 46884046 Ki = 3200 nM T16308 C7J1EI 46884047 Ki = 2300 nM T16308 C3A1CX 46884048 Ki = 1800 nM T16308 CF67NR 46884049 Ki = 13000 nM T16308 CLG36F 46884050 Ki = 3400 nM T16308 CNY23L 46884109 Ki = 2000 nM T16308 CXA3V9 46884110 Ki = 23000 nM T16308 C0IC5D 46884111 IC50 > 50000 nM T16308 CTK27N 46884112 Ki = 2200 nM T16308 CU7J4N 46884113 Ki = 9000 nM T16308 CHW6Z9 46884146 Ki = 3000 nM T16308 C5J1TL 46884147 Ki = 11000 nM T16308 CIB52K 46884148 Ki = 121000 nM T16308 CO2G6S 46884150 Ki = 39000 nM T16308 C2V1YA 46884183 Ki = 11000 nM T16308 CMW52K 46884184 Ki = 4000 nM T16308 CO98ZX 46884185 Ki = 8500 nM T16308 C3IW9C 46884186 Ki = 57000 nM T16308 C1X9FK 46884187 Ki = 53000 nM T16308 C6PU9H 46884230 Ki = 1870 nM T16308 CJ85LK 46884231 Ki = 4430 nM T16308 CD4X1C 46884232 Ki = 7000 nM T16308 CM4D0A 46884233 Ki = 18000 nM T16308 CQAD27 46884263 Ki = 890 nM T16308 C31YMR 46884264 Ki = 3700 nM T16308 CP2A7T 46884265 Ki = 2000 nM T16308 CU1SN0 46884394 IC50 = 31 nM T16308 CIMT25 46884395 IC50 = 1100 nM T16308 CRBG14 46884396 IC50 = 32 nM T16308 CEP3D9 46884397 IC50 = 2500 nM T16308 CI9X6E 46884398 IC50 > 300000 nM T16308 CR0KC6 46884399 IC50 > 300000 nM T16308 CS71XI 46884400 IC50 > 300000 nM T16308 CEAJ15 46906001 Ki = 8 nM T16308 CE20MP 49835937 IC50 = 20000 nM T16308 C1BM2O 49835938 IC50 = 15000 nM T16308 C8FKS7 49835940 IC50 = 4100 nM T16308 CTN37B 49835941 IC50 = 2000 nM T16308 CZ9A7G 50899252 IC50 = 320 nM T16308 CD4W3C 50899253 IC50 = 520 nM T16308 C09GSF 52940692 IC50 = 21000 nM T16308 CWJZ02 52940712 IC50 = 4000 nM T16308 CH20DK 52941817 IC50 = 80000 nM T16308 CMG1S6 52941818 IC50 = 140000 nM T16308 C72WDM 52943237 IC50 = 34000 nM T16308 CU1MV2 52944295 IC50 = 1400 nM T16308 CF71HV 52945544 IC50 = 8000 nM T16308 CR0HJ6 52945672 IC50 = 19000 nM T16308 CO36HS 52946755 IC50 = 220000 nM T16308 CL3V7J 52947957 IC50 = 9400 nM T16308 C6J4OQ 52948352 EC50 = 10000 nM T16308 C8XL6S 52949178 IC50 = 31000 nM T16308 CK2D7U 52952918 IC50 = 2900 nM T16308 C2SI5G 53257623 Ki = 44000 nM T16308 C3L4UW 54580326 Ki = 200 nM T16308 CXR3E1 54580476 IC50 = 9460 nM T16308 C6Z8TP 54581485 IC50 = 16400 nM T16308 C2NO0V 54581486 IC50 = 9810 nM T16308 C2O7MY 54581487 IC50 = 13400 nM T16308 CUF0E5 54581488 IC50 = 5600 nM T16308 CK0IL3 54582488 IC50 > 100000 nM T16308 C7U1LK 54583464 IC50 = 4870 nM T16308 C3KOF4 54583465 IC50 = 9750 nM T16308 CX0FG4 54583466 IC50 = 8500 nM T16308 C02UKH 54584431 IC50 = 9000 nM T16308 CH6U3G 54585390 IC50 = 16400 nM T16308 CM63YQ 54585391 IC50 = 46500 nM T16308 CZ08PE 54586346 IC50 = 33200 nM T16308 C05LVD 54586347 IC50 = 52500 nM T16308 CKE39X 54586348 IC50 = 54200 nM T16308 CD52YW 54587381 IC50 = 23050 nM T16308 CE36MP 54587382 IC50 = 31400 nM T16308 C9UN5S 58243056 IC50 = 2240 nM T16308 CF9DK6 59868882 IC50 > 100000 nM T16308 C4GNS7 60150625 IC50 = 5990 nM T16308 C3TH8K 70681153 IC50 = 18300 nM T16308 CA59OF 70681154 IC50 > 100000 nM T16308 C6JUS7 70681155 IC50 = 54330 nM T16308 C2ZH7I 70683263 IC50 = 10110 nM T16308 CEWJ32 70683264 IC50 = 6310 nM T16308 CKU10X 70687503 IC50 = 11490 nM T16308 C3F4IT 70687504 IC50 = 8930 nM T16308 C8Z6CO 70687505 IC50 = 14520 nM T16308 C1K8RU 70693764 IC50 = 10360 nM T16308 CK0G1O 70695880 IC50 = 53550 nM T16308 CQF25J 71364521 IC50 = 6660 nM T16308 C30DYQ 73346023 IC50 = 600 nM T16308 CKS8M9 73349088 IC50 = 4000 nM T16308 CMC0U7 73355112 IC50 = 6000 nM T16308 C7W3BK 73355113 IC50 = 890 nM T16308 CDEU75 73356684 IC50 = 200 nM T16308 CCQ47X 75039802 IC50 = 4200 nM T16308 CW2GD6 76317298 Ki = 16000 nM T16308 CGP9Y7 76321004 Ki = 15000 nM T16308 CMX5F6 76321005 Ki = 44000 nM T16308 CLJ52Y 76321006 Ki = 32000 nM T16308 CL58FM 86731374 IC50 = 8330 nM T16308 CO5RX8 89486397 IC50 > 100000 nM T16308 CML18X 108137459 IC50 > 100000 nM T16308 CN3GM1 108137463 IC50 > 100000 nM T16308 CZP5B4 108137632 IC50 = 9050 nM T16308 C6VDS3 108137725 IC50 = 22600 nM T16308 CWG5L8 108137732 IC50 = 16550 nM T16308 CA3RG9 114044218 IC50 = 5040 nM T16308 CR14AN 114044219 IC50 = 2520 nM T16308 C3ZJ9G 114044230 IC50 = 4030 nM T16308 CUMS39 118709959 Ki = 173 nM T16308 CF2LC3 118709960 Ki = 189 nM T16308 C5E3SP 118709961 Ki = 780 nM T16308 CJ6D5M 118709962 Ki = 424 nM T16308 C7CD8M 118709963 Ki = 46000 nM T16308 C6R2IK 118709964 Ki = 1000 nM T16308 CX0HI5 118709965 Ki = 10000 nM T16308 CC5AJ7 118709966 Ki = 1900 nM T16308 CK8RA6 118719547 Ki = 400 nM T16308 C7F2YX 118722461 IC50 = 3680 nM T16308 COS7L8 118722462 IC50 > 40000 nM T16308 C8BWJ7 118722463 IC50 = 1470 nM T16308 C3S1CZ 118722464 IC50 > 40000 nM T16308 CNL7E5 118722465 IC50 = 31510 nM T16308 C9U1TV 118722466 IC50 = 830 nM T16308 CBSE31 118722467 IC50 > 40000 nM T16308 CY7OU9 118722468 IC50 = 570 nM T16308 COZR36 118722469 IC50 > 40000 nM T16308 C94TEB 118722470 IC50 = 32300 nM T16308 C7X1WR 118722471 IC50 > 40000 nM T16308 CVF50S 118722472 IC50 = 14110 nM T16308 CLYA60 118722473 IC50 = 2600 nM T16308 C3X7BG 122181534 IC50 = 170 nM T16308 C6N9JD 122194893 IC50 > 100000 nM T16308 CRG92I 122194894 IC50 > 100000 nM T16308 CL1H8Z 122194895 IC50 > 100000 nM T16308 CQAJ92 122194896 IC50 = 39000 nM T16308 CFU7B0 122194897 IC50 > 100000 nM T16308 CB4DM9 122194898 IC50 = 10000 nM T16308 C76ECA 122194899 IC50 > 100000 nM T16308 C3PG9M 122194900 IC50 = 77000 nM T16308 CNJ63H 122194901 IC50 > 100000 nM T16308 C8HG1L 122194902 IC50 > 100000 nM T16308 CD96PL 122194903 IC50 > 100000 nM T16308 CIU95G 122194904 IC50 > 100000 nM T16308 C1CI9G 122194905 IC50 > 100000 nM T16308 C1C2LM 122194906 IC50 > 100000 nM T16308 CF4RE7 122194907 IC50 = 81000 nM T16308 CZ3H7I 122194908 IC50 > 100000 nM T16308 C93LYG 122194909 IC50 > 100000 nM T16308 CY8QP0 122194910 IC50 = 67000 nM T16308 CPY20G 122194911 IC50 = 18000 nM T16308 CE8A1B 122194912 IC50 = 91000 nM T16308 CVL73K 122194913 IC50 = 83000 nM T16308 CJV34R 122194914 IC50 = 91000 nM T16308 C29NFH 122194915 IC50 = 5400 nM T16308 C8VQB5 122194916 IC50 > 100000 nM T16308 CTM3G4 122194917 IC50 > 100000 nM T16308 C3LS6B 122194918 IC50 = 4300 nM T16308 C9L8WA 122194919 IC50 = 19000 nM T16308 C1BR4N 122194920 IC50 > 50000 nM T16308 C48VEQ 122194921 IC50 > 50000 nM T16308 C2AM7R 122194922 IC50 > 100000 nM T16308 CMY1E8 122194923 IC50 = 14000 nM T16308 C0PF2H 122194924 IC50 = 3000 nM T16308 CAC8T0 122194925 IC50 > 100000 nM T16308 C5LZJ8 137633418 IC50 = 1070 nM T16308 C6FV1K 137634154 IC50 = 3570 nM T16308 CXO62Z 137635918 IC50 = 2310 nM T16308 CIHV78 137636151 IC50 > 10000 nM T16308 CGIE74 137638055 IC50 > 10000 nM T16308 CF6MI7 137639703 IC50 = 3800 nM T16308 CD8B4M 137641636 IC50 = 2820 nM T16308 CY3BK4 137644555 IC50 = 1060 nM T16308 C2AEI9 137646424 IC50 = 2100 nM T16308 CB1I3P 137647067 IC50 = 4290 nM T16308 CQ8I1F 137652908 IC50 = 9600 nM T16308 CH2J1K 137656019 IC50 > 10000 nM T16308 CG9SV0 137656633 IC50 = 1330 nM T16308 CY1AB9 137656969 IC50 > 10000 nM T16308 C7J2WV 137657062 IC50 > 10000 nM T16308 C9WP6I 137660249 IC50 = 2350 nM T16308 C1CNH9 137661852 IC50 = 4790 nM T16308 CNXY47 138454795 IC50 = 874 nM T16308 CRD72V 141483210 IC50 = 1870 nM T16308 CHU1K4 141483211 IC50 = 470 nM T16308 CQ10JV 141483212 IC50 = 1100 nM T16308 CQ1I8F 141483217 IC50 = 1020 nM T16308 C7RGL9 141483219 IC50 = 18680 nM T16308 CFH0C7 141483224 IC50 = 2200 nM T16308 CMC79W 141483227 IC50 = 720 nM T16308 CM7CL9 141483233 IC50 = 11280 nM T16308 CX4KF9 141483235 IC50 = 1890 nM T16308 C0I1EM 141483240 IC50 = 13890 nM T16308 CNJ40T 141483241 IC50 = 13620 nM T16308 C5LH6N 145967653 IC50 > 100000 nM T16308 C7VNA0 145967916 IC50 = 7280 nM T16308 CZS8U1 145967923 IC50 = 2170 nM T16308 CQR6E8 145968164 IC50 > 100000 nM T16308 CEJ1S2 145968301 IC50 > 100000 nM T16308 C4JA3L 145968650 IC50 = 13870 nM T16308 C2SPC5 145968765 IC50 = 4080 nM T16308 C6O0VF 145968864 IC50 > 100000 nM T16308 CL1YA7 145969010 IC50 > 100000 nM T16308 CE07JF 145969015 IC50 = 1680 nM T16308 CO40SQ 145969074 IC50 > 100000 nM T16308 CO9W6Z 145969565 IC50 > 100000 nM T16308 CJMB97 145969756 IC50 = 4360 nM T16308 C9XK5M 145970008 IC50 > 100000 nM T16308 CS3P2G 145970114 IC50 = 9870 nM T16308 C2TQ4E 145970180 IC50 = 7270 nM T16308 C1VO8C 145970188 IC50 > 100000 nM T16308 CT0FV8 145970386 IC50 = 34040 nM T16308 CN4L9X 145970621 IC50 = 33500 nM T16308 CA8WO6 145971036 IC50 = 20200 nM T16308 C2O8ED 145971130 IC50 > 100000 nM T16308 C9TZ6K 145971175 IC50 > 100000 nM T16308 CL1G9E 145981256 IC50 = 2180 nM T16308 C75LXF 145981632 IC50 = 550 nM T16308 CJ5P8L 145983687 IC50 = 1580 nM T16308 CQP4A7 145986584 IC50 = 26670 nM T16308 CXE9Q6 145987041 IC50 = 18900 nM T16308 C7F4MC 145988608 IC50 = 2680 nM T16308 C5XY8U 145988732 IC50 = 1270 nM T16308 C3I4KC 145988830 IC50 = 3480 nM T16308 C14XBZ 145989474 IC50 = 5200 nM T16308 C3WVO1 145990332 IC50 = 460 nM T16308 C64WLQ 145990695 IC50 = 970 nM T16308 CZF7X6 145992067 IC50 = 1010 nM T16308 CD6HL8 145993842 IC50 = 680 nM T16308 CPI68O 155516500 IC50 = 19720 nM T16308 CH0CS6 155517460 IC50 = 1000 nM T16308 CC1HR5 155520254 IC50 > 100000 nM T16308 CYF04X 155524668 IC50 = 2260 nM T16308 CC1E0B 155525657 IC50 = 2890 nM T16308 CMY62G 155532089 Ki = 1370 nM T16308 CY3RB9 155533153 IC50 = 9810 nM T16308 C90IEM 155536416 Ki = 5470 nM T16308 C1TS6Y 155538914 IC50 = 7560 nM T16308 CHLD92 155547270 IC50 = 7830 nM T16308 C4F2PA 155554836 IC50 = 3570 nM T16308 CQ83OH 155558997 IC50 = 7270 nM T16308 C5G9VX 155561107 IC50 = 330 nM T16308 CTCE89 155561370 IC50 = 5400 nM T16308 CV5QU1 155561997 IC50 = 1530 nM T16308 C4QTW6 155566014 IC50 > 100000 nM T16308 D02XEX 11168203 IC50 = 50360 nM T16308 D06ZWX 6197 Ki > 200000 nM T16308 D07UCF 615184 IC50 = 6100 nM T16308 D08MJE 45100499 Ki = 1800 nM T16308 D08TZA 46884149 Ki = 17000 nM T16308 D0M9FC 46884013 Ki = 9700 nM T16308 D0N9NS 46884012 Ki = 2800 nM T16308 D0Q9YG 46884229 Ki = 12800 nM T16308 D0U8IF 10114 IC50 > 10000 nM T16308 D0W4CN 44409555 Ki = 18.3 nM T16308 D0W8MX 44409591 Ki = 547 nM T16308 D0XF6C 2738139 IC50 = 180000 nM T16308 D0Y7PY 44409592 Ki = 258 nM T61518 D02XNW 5494449 IC50 = 420 nM T61518 D03HUX 49792852 IC50 = 744 nM T61518 D04UUD 10430360 IC50 = 340 nM T61518 D05PZB 135398495 IC50 = 685 nM T61518 D08FIX 135398499 IC50 = 0.41 nM T61518 D0E3TC 44259 IC50 = 0.542 nM T61518 D0O0LS 25141092 IC50 > 10000 nM T61518 C4DW3Y 660621 IC50 = 1185 nM T61518 C3GHQ1 690227 IC50 > 5000 nM T61518 CIZ9D2 2216908 IC50 > 5000 nM T61518 CJAQ19 2491127 IC50 = 388 nM T61518 C1OW6X 3141330 IC50 > 5000 nM T61518 CF7HW1 3620985 IC50 = 400 nM T61518 CA3C5S 3685259 IC50 = 180 nM T61518 CB7WK3 5938113 IC50 = 1400 nM T61518 CV50PJ 12451684 IC50 = 6100 nM T61518 CJ8W9Z 16044323 IC50 > 5000 nM T61518 C3P8XU 16760499 IC50 = 440 nM T61518 C46DEZ 17816913 IC50 > 20000 nM T61518 CRAH02 42647778 IC50 > 5000 nM T61518 C9WL5N 42647801 IC50 > 5000 nM T61518 CBI04W 42647935 IC50 = 1116 nM T61518 CSP6D8 43831079 IC50 = 4126 nM T61518 C1U7PZ 43831080 IC50 = 1774 nM T61518 C3VRO9 44557921 IC50 > 10000 nM T61518 CLS29B 46872626 IC50 > 10000 nM T61518 C6J4OP 47001335 IC50 = 192 nM T61518 CF91RS 49843531 IC50 > 10000 nM T61518 C2Y6QS 50938552 IC50 > 10000 nM T61518 C9NYP4 51036677 IC50 > 10000 nM T61518 C4WRY3 51037112 IC50 > 10000 nM T61518 CRI28Z 51037948 IC50 > 10000 nM T61518 CV13QY 58540422 IC50 > 10000 nM T61518 CMO15Y 63901349 IC50 = 160000 nM T61518 CV63UL 67240318 IC50 > 10000 nM T61518 CCN01X 71547862 IC50 > 10000 nM T61518 C6R8DI 72943374 IC50 = 258 nM T61518 C4U5NV 73442760 IC50 = 37 nM T61518 CGDB30 74538658 IC50 = 19 nM T61518 CGJ0Q3 78350436 IC50 = 2100 nM T61518 C27SIH 78350438 IC50 = 31000 nM T61518 CGKW40 78350469 IC50 = 3100 nM T61518 C6FR9J 78350471 IC50 = 4200 nM T61518 CS4A3I 78673829 IC50 = 1000 nM T61518 C7QSR8 85325330 IC50 = 520 nM T61518 C0NR6S 85325332 IC50 = 650 nM T61518 CY0UC4 90645194 IC50 > 10000 nM T61518 CY7BI2 118706214 IC50 > 10000 nM T61518 C6S4XB 118720606 IC50 = 410 nM T61518 C2K6LE 118720607 IC50 = 24000 nM T61518 C06LWS 118720608 IC50 = 5100 nM T61518 CS4I7U 118720609 IC50 = 7.6 nM T61518 C75PHN 119058124 IC50 = 2 nM T61518 CJ6FQ7 119058125 IC50 = 410 nM T61518 CWDX84 119058126 IC50 = 13 nM T61518 C5YJ9E 122705889 IC50 = 900 nM T61518 CS2E6X 127048234 IC50 = 5000 nM T61518 C2YHT0 127048915 IC50 = 670 nM T61518 CF0KU7 127050847 IC50 = 520 nM T61518 C24DQX 127051101 IC50 = 64 nM T61518 CH1YA6 127051102 IC50 = 80 nM T61518 C1Y2GO 127051103 IC50 = 1 nM T61518 CP73XR 127051104 IC50 = 25 nM T61518 CCZH52 127051105 IC50 = 260 nM T61518 C6LNW2 127052230 IC50 = 4 nM T61518 CR48OV 127052231 IC50 = 36 nM T61518 CS59XH 127052232 IC50 = 210 nM T61518 CW8Z6C 127052233 IC50 = 0.3 nM T61518 C2AN7T 134611886 IC50 > 100000 nM T61518 CJI0G1 135520135 IC50 = 2800 nM T61518 CHA4N2 136013680 IC50 > 10 nM T61518 CH64ID 136175114 IC50 > 10000 nM T61518 C1YUD0 136219394 IC50 > 10 nM T61518 COG2M5 136242661 Ki = 0.47 nM T61518 CIU8W3 136254389 IC50 > 10 nM T61518 CSGM03 137210056 IC50 = 1000 nM T61518 C04YDK 137248544 Ki = 0.39 nM T61518 C2J5CN 137293686 Ki = 2.3 nM T61518 C97CMT 137293687 Ki = 358 nM T61518 CDB68K 137293702 Ki > 650 nM T61518 CRYI28 137293705 Ki = 3.1 nM T61518 CMB78I 137301774 Ki = 0.68 nM T61518 CHF1V3 137301775 Ki = 46 nM T61518 C0W3KM 137631515 IC50 = 120 nM T61518 C2Z6PU 137632011 IC50 = 3500 nM T61518 C6VKD9 137633401 IC50 = 9.2 nM T61518 CU75HC 137633476 IC50 = 3700 nM T61518 CT41DA 137636064 IC50 = 400 nM T61518 CYH3P1 137636760 IC50 = 6800 nM T61518 CFYB36 137638498 Ki = 8.8 nM T61518 CGP48Y 137639114 IC50 = 1.5 nM T61518 CNU81W 137641500 IC50 = 8.8 nM T61518 C6G5BQ 137642064 IC50 = 8900 nM T61518 CJ4MI7 137642078 IC50 = 1.1 nM T61518 CZ3C1M 137643225 IC50 = 720 nM T61518 CINF50 137644022 IC50 = 2600 nM T61518 C4U9QF 137646381 IC50 = 1300 nM T61518 CMZ02P 137649794 IC50 = 0.15 nM T61518 C1KO7R 137651632 IC50 = 2100 nM T61518 CP04RX 137652802 IC50 = 740 nM T61518 C5MG7R 137653946 IC50 = 1.5 nM T61518 CM9H2O 137655933 IC50 = 12 nM T61518 C40GAX 137659707 IC50 = 7700 nM T61518 CR2OA8 155510507 IC50 = 141 nM T61518 C2MD1Q 155513187 IC50 > 10000 nM T61518 C2WGR6 155518450 IC50 > 5000 nM T61518 CZ3RW5 155521164 IC50 = 112 nM T61518 CTXD61 155522409 IC50 = 222 nM T61518 C01QHJ 155522952 IC50 = 122 nM T61518 CP8A0W 155523587 IC50 = 599 nM T61518 CHQ63Z 155531664 IC50 = 638 nM T61518 C8OL9Y 155532496 IC50 = 1701 nM T61518 C0AR4Z 155533016 IC50 > 5000 nM T61518 CDZ18P 155535001 IC50 = 241 nM T61518 CR9G3K 155538487 IC50 = 540 nM T61518 CB01CY 155540962 IC50 = 707 nM T61518 CAYF68 155543222 IC50 = 269 nM T61518 C1KBH2 155547976 IC50 = 350 nM T61518 C19QDP 155549136 IC50 = 575 nM T61518 C0STI2 155549197 IC50 > 5000 nM T61518 CH3K7T 155552256 IC50 > 5000 nM T61518 CHE7F8 155554129 IC50 = 1417 nM T61518 CN4TI9 155555255 IC50 = 98 nM T61518 CHU10X 155558521 IC50 > 5000 nM T61518 CE4LF2 155558943 IC50 = 313 nM T61518 CG4HQ6 155559449 IC50 > 5000 nM T61518 CUW59T 155559912 IC50 = 1353 nM T61518 CT5W1V 155566733 IC50 = 494 nM T61518 D05GMB 135461425 Ki = 149 nM T61518 D09HVH 135566652 IC50 > 10 nM T61518 D09LPL 5329103 IC50 = 760 nM T61518 D0IR6U 5494425 IC50 = 330 nM T10265 D05MQK 110635 IC50 > 50000 nM T10265 D07ESC 11561674 IC50 = 24 nM T10265 D09QEI 4740 IC50 > 90000 nM T10265 D0F8RA 2153 IC50 > 200000 nM T10265 D0R4UW 449193 Ki = 0.3981 nM T10265 D0Z7ZM 135398744 IC50 = 20000 nM T10265 D00JED 24806574 IC50 = 240 nM T10265 D03QJL 3671 IC50 = 65 nM T10265 D09TFB 9896267 IC50 = 13 nM T10265 D0IZ8X 90111638 IC50 = 2013 nM T10265 D0M7CB 9919680 IC50 = 5.1 nM T10265 D0SM0W 44591583 IC50 = 55 nM T10265 D0T5PO 5092 IC50 = 34 nM T10265 D0Z2FB 154575 IC50 = 0.041 nM T10265 D00YPW 135399235 Ki > 50000 nM T10265 D01FXD 9802841 IC50 = 60 nM T10265 D02EMR 151170 IC50 = 25 nM T10265 D07FHZ 5087 Ki = 1930 nM T10265 D08SNX 135430158 Ki = 270 nM T10265 D0BK6B 3021729 Ki > 50000 nM T10265 D0F0CS 5723 IC50 = 1410 nM T10265 D0H9KW 9578243 IC50 = 960 nM T10265 D0I0GM 449190 IC50 = 420 nM T10265 D0U7PS 9827968 IC50 < 0.01 nM T10265 D0UG4T 127928 IC50 = 1.4 nM T10265 C8GAZ7 8394 IC50 = 520 nM T10265 C4B3YS 78864 IC50 = 231 nM T10265 C1H8NR 155248 IC50 = 18100 nM T10265 C52SNB 180510 IC50 = 44000 nM T10265 CYWS98 185848 IC50 = 4500 nM T10265 C73SFB 266817 IC50 = 3530 nM T10265 C63TBQ 314892 IC50 = 15.85 nM T10265 CP3Y7O 656968 IC50 = 56 nM T10265 C29DYI 656969 IC50 = 33 nM T10265 C1B6ZL 662965 IC50 = 540 nM T10265 CM0Q1K 675863 IC50 = 1258.93 nM T10265 CZN6S9 743974 IC50 > 25118.86 nM T10265 CM86KB 826384 IC50 = 190 nM T10265 CR35EF 832190 IC50 = 6700 nM T10265 COS03W 1204288 IC50 = 17900 nM T10265 CK8DT9 1205767 IC50 = 6910 nM T10265 C3D0HY 1232680 IC50 = 6510 nM T10265 CPXC25 1368101 IC50 = 5300 nM T10265 C9H6YT 1390827 IC50 = 64820 nM T10265 CC82DS 1418559 IC50 = 54650 nM T10265 C8G2PE 1506612 IC50 = 3500 nM T10265 CWJS81 1539584 IC50 = 14100 nM T10265 C8GCU4 2145707 IC50 = 740 nM T10265 CO2C9B 2170892 IC50 = 11200 nM T10265 CLX0W5 2566813 IC50 = 12100 nM T10265 CW57NL 2852188 IC50 = 50.12 nM T10265 CY7IG8 2853935 IC50 = 630.96 nM T10265 CVJ36Q 2862736 IC50 > 2511.89 nM T10265 C4LSR7 2886111 IC50 = 199.53 nM T10265 C4H9EN 3058801 Ki = 447 nM T10265 CJC7M6 3604361 IC50 = 79.43 nM T10265 CHV64Q 3713518 IC50 = 26 nM T10265 CQLN58 3826564 IC50 = 5000 nM T10265 CV0AQ4 4198517 IC50 = 3710 nM T10265 C7HST8 4231279 IC50 = 1995.26 nM T10265 CL1Q4X 4254532 IC50 = 5.7 nM T10265 CT8YE5 4316226 IC50 = 90 nM T10265 CB73HU 4398380 IC50 = 10 nM T10265 C12SRB 5214710 IC50 = 25.12 nM T10265 CFJ62Y 9799389 IC50 = 34 nM T10265 CYXD04 9810934 IC50 = 8 nM T10265 CRT85L 9821178 IC50 = 3.162 nM T10265 CL70YN 9840066 IC50 = 2.1 nM T10265 C5YQB0 9859898 IC50 = 40000 nM T10265 CR01PJ 9865970 IC50 = 400 nM T10265 CAY84B 9869820 IC50 = 0.85 nM T10265 CIT6P8 9876393 IC50 = 0.631 nM T10265 CJG9R8 9904574 IC50 = 1600 nM T10265 CCPY51 9908333 IC50 = 19 nM T10265 C76RTB 9924539 IC50 = 34 nM T10265 CZM42J 9926935 IC50 = 486 nM T10265 CA42XV 9948833 IC50 = 24.1 nM T10265 CT14LN 9972167 IC50 = 63.1 nM T10265 CMH2J5 9972313 Ki = 426.58 nM T10265 CGE8T2 9975276 IC50 < 10 nM T10265 C8ZX0U 9976104 Ki = 67.61 nM T10265 CI6UN2 9995212 Ki = 181.97 nM T10265 CV6TO1 9995407 IC50 = 17.9 nM T10265 COW3G0 9997331 Ki = 281.84 nM T10265 CA9YF5 9998837 IC50 = 168 nM T10265 CFPR64 9999276 IC50 = 49 nM T10265 C53HZC 9999401 IC50 = 1333 nM T10265 CA0XZ7 10000779 Ki = 60.26 nM T10265 C4ZKB5 10019613 Ki = 269.15 nM T10265 C70PEG 10022725 Ki = 33.88 nM T10265 CX1YH0 10023563 Ki = 158.49 nM T10265 C3A6RV 10027487 IC50 = 0.57 nM T10265 CN7HJ5 10039641 Ki = 89.13 nM T10265 CCA82X 10043075 IC50 = 158.49 nM T10265 CAM0J5 10043254 Ki = 741.31 nM T10265 C1N7GA 10045809 IC50 = 19 nM T10265 C1W2BY 10064555 Ki = 58.88 nM T10265 CG4AV5 10068352 Ki = 426.58 nM T10265 CL63VR 10087314 Ki = 186.21 nM T10265 C2S1WA 10088201 Ki = 70.79 nM T10265 C8T3LV 10090103 IC50 = 615 nM T10265 C3G2UF 10090751 IC50 = 19.95 nM T10265 C6T4JS 10091127 IC50 = 1333 nM T10265 CK2ST7 10091864 Ki = 50 nM T10265 CK5C9Z 10119563 IC50 = 0.3 nM T10265 C1EVS3 10119564 IC50 = 0.4 nM T10265 C83BSD 10128917 IC50 = 0.1 nM T10265 CWDR26 10129145 IC50 = 0.6 nM T10265 CME68G 10152836 IC50 = 140 nM T10265 C0PVT2 10153372 IC50 = 210 nM T10265 C7D5IT 10158829 IC50 = 43 nM T10265 CBT4P1 10177031 IC50 = 20 nM T10265 C3X9DK 10183196 IC50 = 6.4 nM T10265 CUXV40 10183769 IC50 = 0.3 nM T10265 CY9HS7 10185841 IC50 = 0.07 nM T10265 CVUZ36 10195164 IC50 = 3 nM T10265 C8LYH6 10196396 IC50 = 0.3 nM T10265 CSQ16M 10196596 IC50 = 0.1 nM T10265 CTV6F9 10196609 IC50 = 0.1 nM T10265 CTZ7Q8 10196916 IC50 = 0.3 nM T10265 CZG54F 10197046 IC50 = 250 nM T10265 CE5LH4 10199681 IC50 = 17 nM T10265 C61CZK 10205978 IC50 = 19 nM T10265 CPU09I 10210579 IC50 = 0.5 nM T10265 C8JR4W 10221093 IC50 = 9000 nM T10265 CX9LV3 10232106 IC50 = 1.1 nM T10265 CH3Y8I 10245392 Ki = 109.65 nM T10265 CFDH45 10245470 Ki = 154.88 nM T10265 CX0BK5 10246197 Ki = 144.54 nM T10265 CI5Y3F 10254618 IC50 = 0.88 nM T10265 C2KBI9 10266977 Ki = 89.13 nM T10265 CB16GD 10267029 IC50 = 251.19 nM T10265 C7RH4B 10270013 IC50 = 156 nM T10265 C48ENU 10289786 IC50 = 4.2 nM T10265 CT5FL2 10289848 IC50 = 0.03 nM T10265 CECW14 10301548 IC50 = 0.2 nM T10265 C5IF9A 10312566 IC50 = 0.4 nM T10265 CY74PB 10335857 Ki = 63 nM T10265 CR73QT 10336025 IC50 = 15.85 nM T10265 C30JKP 10338622 Ki = 30 nM T10265 CJ7YZ9 10345293 IC50 = 0.54 nM T10265 C35IAZ 10358514 Ki = 758.58 nM T10265 C0QKV3 10360335 Ki = 45.71 nM T10265 CY9FX2 10381125 Ki = 70 nM T10265 CFH73T 10406734 Ki = 56.23 nM T10265 CER6Z4 10424262 IC50 = 25.12 nM T10265 CT7CP0 10429315 Ki = 70.79 nM T10265 C9A1JH 10432102 IC50 = 225 nM T10265 CL3NZ6 10448469 IC50 = 10 nM T10265 C4ME8I 10449388 Ki = 316.23 nM T10265 C83XZL 10451240 Ki = 588.84 nM T10265 CD09NL 10451631 IC50 = 187 nM T10265 CAK2Q1 10452194 IC50 = 9.2 nM T10265 CI7Y3L 10467846 Ki = 5888.44 nM T10265 C0C6VT 10471954 Ki = 158.49 nM T10265 CBK9N4 10472881 Ki = 64.57 nM T10265 CXWB17 10475192 IC50 = 7.943 nM T10265 CC1BU8 10543370 Ki = 338 nM T10265 CF48IV 10615343 Ki = 27 nM T10265 C9CLS3 10639193 Ki = 282 nM T10265 CDH2P7 10686898 Ki = 583 nM T10265 C0A7DI 11017241 IC50 = 40 nM T10265 CUY0M5 11153991 IC50 = 25.12 nM T10265 C3B1QP 11161553 IC50 = 13000 nM T10265 C71WZV 11164397 IC50 = 31.62 nM T10265 CU1ZY7 11213333 IC50 = 2.512 nM T10265 C6WUB7 11225327 IC50 = 0.01995 nM T10265 C9B4AY 11269083 IC50 = 2.512 nM T10265 C6VL4T 11280182 IC50 = 3.981 nM T10265 C3TQ2G 11293791 IC50 = 0.1 nM T10265 CATL36 11304132 IC50 = 0.7943 nM T10265 C8SKJ6 11314577 IC50 = 19.95 nM T10265 C7T4XK 11350199 IC50 = 0.3162 nM T10265 C46XUS 11394750 IC50 = 15.85 nM T10265 CNU8E6 11397103 IC50 = 0.1259 nM T10265 CZS96V 11406358 IC50 = 0.3981 nM T10265 C46VGX 11406619 IC50 = 31.62 nM T10265 CSVI94 11430281 IC50 = 3.162 nM T10265 C45VZC 11438405 IC50 > 16000 nM T10265 CNV60P 11449090 IC50 > 30000 nM T10265 CG37OU 11511603 IC50 = 95 nM T10265 CQ8G9F 11525525 IC50 = 3.8 nM T10265 C3MVD1 11525902 IC50 = 284 nM T10265 CS5U1Z 11532316 IC50 = 45 nM T10265 C6UMB2 11532832 IC50 = 8.05 nM T10265 CKD51J 11540543 IC50 = 167 nM T10265 C7FQU3 11545707 IC50 = 1 nM T10265 CX0FM3 11547713 IC50 = 0.6 nM T10265 C0EZ7X 11555069 IC50 = 3697 nM T10265 C8R1NX 11566058 IC50 = 42 nM T10265 CUBT56 11576136 IC50 = 1765 nM T10265 C5V0RU 11584000 IC50 = 213 nM T10265 CHU90R 11598626 IC50 = 0.06 nM T10265 C3G1BO 11604203 IC50 = 1790 nM T10265 CN6B3P 11612979 IC50 = 1198 nM T10265 C1G3EI 11620160 IC50 = 2.6 nM T10265 CE24AU 11626787 IC50 = 22 nM T10265 C0BD7Q 11628421 IC50 = 4.5 nM T10265 C37TWP 11633996 IC50 = 3.6 nM T10265 C6GY9D 11635241 IC50 = 1 nM T10265 COLF16 11639342 IC50 = 1900 nM T10265 C8U5VK 11641556 IC50 = 2.9 nM T10265 C8EX6Z 11648288 IC50 = 11 nM T10265 C83NLR 11648915 IC50 = 21 nM T10265 CXD82O 11649109 IC50 = 0.6 nM T10265 CX2ZD7 11650267 Ki = 199 nM T10265 CFM64H 11662453 IC50 = 7.2 nM T10265 CR8CQ7 11669507 IC50 = 2550 nM T10265 CQPW60 11705339 IC50 = 2.9 nM T10265 C0I5BW 11711290 IC50 = 37 nM T10265 CVJ10R 11713455 IC50 = 13 nM T10265 C0FC4T 11719711 IC50 = 274 nM T10265 CLEK64 11726110 Ki = 30.2 nM T10265 CK9F0W 11741974 Ki = 181.97 nM T10265 CA26IK 11742611 IC50 = 20 nM T10265 CW6A8Y 11742832 Ki = 30 nM T10265 C4Z9EM 11750855 IC50 = 1.585 nM T10265 CROY49 11754228 IC50 = 0.54 nM T10265 CC92YE 11755033 IC50 = 0.53 nM T10265 C7AP8V 11778917 Ki = 91.2 nM T10265 CM57TH 11779811 Ki = 100 nM T10265 C54KPM 11794796 Ki = 550 nM T10265 C8YRP7 11955134 IC50 = 470 nM T10265 CG3RA6 11955200 IC50 = 42 nM T10265 C1B4XD 11992634 IC50 = 290 nM T10265 CPX16N 11993169 IC50 > 2000 nM T10265 C1A2IB 12001199 IC50 = 707.95 nM T10265 CL2FY7 15192730 Ki = 160 nM T10265 C40KZA 15434926 IC50 = 210 nM T10265 C4ESY5 15942639 IC50 = 0.2 nM T10265 C07XUL 15950810 IC50 = 68 nM T10265 CN3I4Z 15950948 IC50 = 19 nM T10265 C3BI9R 15951010 IC50 = 32 nM T10265 CWH1A8 15951076 IC50 = 15 nM T10265 C6VN5F 16067799 IC50 = 6 nM T10265 CPQE51 16067902 IC50 = 337 nM T10265 CF3U9Y 16067903 IC50 = 235 nM T10265 CD50HG 16067905 IC50 = 79 nM T10265 CMB3Z5 16067906 IC50 = 0.1 nM T10265 C31LJY 16103072 IC50 = 430 nM T10265 C2YI5D 16230554 IC50 = 46100 nM T10265 CMN23R 16391719 IC50 = 14000 nM T10265 CYN39I 16666580 IC50 = 410 nM T10265 C0HI2G 16666581 IC50 = 79 nM T10265 CAW98T 16666618 IC50 = 15 nM T10265 CD1VU8 16666619 IC50 = 35 nM T10265 CJP10M 16666620 IC50 = 7.5 nM T10265 CM91TF 16666621 IC50 = 150 nM T10265 C4U3WX 16666622 IC50 = 110 nM T10265 COG39H 16727125 IC50 = 0.5 nM T10265 CQ5XC2 17436003 IC50 = 15000 nM T10265 CF72AG 17559143 IC50 = 26000 nM T10265 CXFT59 17757146 IC50 = 37.2 nM T10265 CBX29P 17989733 IC50 = 93 nM T10265 C1PZ8C 18734933 IC50 = 185 nM T10265 C9DE6Y 20814950 IC50 = 1.8 nM T10265 C9B5XO 21823929 IC50 = 630.96 nM T10265 CTY8Q2 21823948 IC50 = 158.49 nM T10265 C3M5NF 21865580 IC50 = 200 nM T10265 C4CWR6 21865595 IC50 = 4000 nM T10265 C6T5NZ 21865599 IC50 = 400 nM T10265 CULE52 21865620 IC50 = 90 nM T10265 CINH54 21865627 IC50 = 0.5 nM T10265 CMHF08 22083604 IC50 = 1.1 nM T10265 C34FLM 22083724 IC50 = 0.3 nM T10265 CWIT18 22083784 IC50 = 0.3 nM T10265 CKP50C 22337156 IC50 = 263 nM T10265 CM9RX0 22337173 IC50 = 520 nM T10265 CR4T9J 22337182 Ki = 250 nM T10265 CFAQ86 22343616 IC50 = 6600 nM T10265 CC1Z3A 22456843 IC50 = 85.8 nM T10265 CTU51Z 22456845 IC50 = 367 nM T10265 C5TQ0N 22456850 IC50 = 341 nM T10265 CD48PX 23218492 IC50 = 22.2 nM T10265 CDNX73 23649292 IC50 = 45 nM T10265 CJ0ZF1 24180492 IC50 = 19 nM T10265 CAJ57O 24751843 IC50 = 114000 nM T10265 CR0D6X 24751988 IC50 = 16000 nM T10265 CL79TD 24751991 IC50 = 29000 nM T10265 CO15XH 24752867 IC50 = 4.9 nM T10265 C7QEC1 24772445 IC50 = 0.51 nM T10265 C1H2XW 24772446 IC50 = 10 nM T10265 CHX26Y 24772447 IC50 = 7 nM T10265 CJSX90 24772448 IC50 = 110 nM T10265 CZ4ID6 24772449 IC50 = 2.8 nM T10265 CP5R8O 24772450 IC50 = 13 nM T10265 C2LS4C 24772511 IC50 = 4.1 nM T10265 C51NQP 24772512 IC50 = 31 nM T10265 CDU9R1 24772513 IC50 = 8 nM T10265 C1PI8A 24772514 IC50 = 0.2 nM T10265 CZF02U 24798187 IC50 = 15 nM T10265 C07DBW 24798271 IC50 = 9.4 nM T10265 CHB7O2 24798272 IC50 = 2.9 nM T10265 CVE1K5 24798273 IC50 = 5.5 nM T10265 C2ET7F 24799903 IC50 = 1070 nM T10265 C0GHB4 24799905 IC50 = 150 nM T10265 CY9H4A 24799906 IC50 = 63 nM T10265 C3TJ2G 24799907 IC50 = 200 nM T10265 C7ZH3R 24800081 IC50 = 690 nM T10265 CM9DG6 24800082 IC50 = 360 nM T10265 C0UY9O 24802801 IC50 = 300 nM T10265 C73ABX 24802803 IC50 = 1010 nM T10265 C0LEU9 24802804 IC50 = 21 nM T10265 CA74HQ 24804333 IC50 = 3 nM T10265 CJGZ93 24804334 IC50 = 0.5 nM T10265 C20JRY 24804335 IC50 = 0.2 nM T10265 CG64YI 24804336 IC50 = 1.7 nM T10265 C39PBK 24804498 IC50 = 2.2 nM T10265 CK74LY 24841825 IC50 = 0.631 nM T10265 CS6KQ0 24849255 IC50 = 5 nM T10265 C57WUF 24849256 IC50 = 3 nM T10265 CK2IF5 24849257 IC50 = 2 nM T10265 CKW6Q3 24849380 IC50 = 5 nM T10265 C3SZG2 24849572 IC50 = 21 nM T10265 CSY6G1 24849618 IC50 = 1 nM T10265 CXJC34 24849668 IC50 = 1180 nM T10265 CJA9R5 24849669 IC50 = 80 nM T10265 CVD5B0 24849709 IC50 = 43 nM T10265 C8YH4E 24849714 IC50 = 5 nM T10265 CG8Z2I 24849846 IC50 = 17 nM T10265 C8DC2M 24849847 IC50 = 2 nM T10265 CJX2G7 24849885 IC50 = 2 nM T10265 C64GKY 24957666 IC50 = 2300 nM T10265 C4QJ2S 24958040 IC50 = 500 nM T10265 CW8YM2 24958042 IC50 = 16000 nM T10265 CAO1H6 24958416 IC50 = 3300 nM T10265 CMT36Y 24958421 IC50 > 30000 nM T10265 C6EQG2 24963293 IC50 > 2000 nM T10265 C9TS3H 25018106 IC50 = 280 nM T10265 CPIO29 25018348 IC50 = 430 nM T10265 C2B4NM 25026184 IC50 = 0.6 nM T10265 C8YBW4 25055989 IC50 = 160 nM T10265 CC58QZ 25055991 IC50 = 2930 nM T10265 CBL3C7 25056255 IC50 = 17 nM T10265 CB79EW 25056256 IC50 = 50 nM T10265 C7V4AS 25142306 IC50 = 6.7 nM T10265 C1MCK3 25142307 IC50 = 0.38 nM T10265 C4J0YD 25196719 IC50 = 8730 nM T10265 C4APQ0 25596969 IC50 = 16000 nM T10265 CTQI51 26273258 IC50 = 7400 nM T10265 CLKF86 27351067 IC50 > 1000 nM T10265 CN4W2U 27659581 IC50 = 15800 nM T10265 CN1QG6 27659634 IC50 = 51600 nM T10265 C5Q0IN 42647289 IC50 = 2.9 nM T10265 CNIE98 44143458 IC50 = 1.6 nM T10265 CW8OB3 44243146 Ki > 10000 nM T10265 C1UDI7 44284299 Ki = 794.33 nM T10265 CZY71A 44284318 Ki = 194.98 nM T10265 CCO40U 44302055 Ki = 190 nM T10265 CG4DR8 44302271 Ki = 1570 nM T10265 CGCI15 44302290 Ki = 1470 nM T10265 C60ASC 44302299 Ki = 4420 nM T10265 CS64YP 44302300 Ki = 290 nM T10265 CRFQ73 44302318 Ki = 80 nM T10265 C8H5KB 44302319 Ki = 150 nM T10265 CH7B2U 44302345 Ki = 50 nM T10265 C1HY2N 44302362 Ki = 1130 nM T10265 CLD6S9 44302363 Ki = 40 nM T10265 CT6V7I 44302374 Ki = 60 nM T10265 C4XFM5 44302392 Ki = 350 nM T10265 CH24DK 44302395 Ki = 1880 nM T10265 C81UZW 44302421 Ki = 4630 nM T10265 C2EFA6 44302457 Ki = 2290 nM T10265 CI7T5U 44302569 Ki = 240 nM T10265 CZS34P 44302570 Ki = 1200 nM T10265 CHL81S 44302582 Ki = 80 nM T10265 CTZ4F3 44302604 Ki = 14400 nM T10265 C7AY0R 44302614 Ki = 1570 nM T10265 CI2X6K 44302636 Ki = 380 nM T10265 C1T4FM 44302642 Ki = 1480 nM T10265 C38QZM 44302662 Ki = 810 nM T10265 C97EXY 44302664 Ki = 6030 nM T10265 C2SLH8 44324331 IC50 = 10.9 nM T10265 C6TM8Z 44372695 IC50 = 21 nM T10265 CA1MV5 44372706 IC50 = 28.4 nM T10265 C5HVW8 44372709 IC50 = 241 nM T10265 C5OYN4 44372911 IC50 = 22.4 nM T10265 C9UFG2 44372973 IC50 > 1000 nM T10265 C0G9MH 44373061 IC50 = 36.1 nM T10265 C9HD1E 44373136 IC50 = 196 nM T10265 C1WAI9 44373180 IC50 = 56.5 nM T10265 C9XPC1 44373185 IC50 = 67.6 nM T10265 C92XAF 44373203 IC50 = 30 nM T10265 C54WVS 44373279 IC50 = 109.6 nM T10265 C1S2WR 44373280 IC50 = 277 nM T10265 CX05SR 44373291 IC50 > 1000 nM T10265 CH9Q5Z 44373305 IC50 = 327 nM T10265 CF0JM6 44373307 IC50 = 24.3 nM T10265 C4W0IU 44373457 IC50 = 39.2 nM T10265 CI6X0L 44373488 IC50 = 399 nM T10265 CLMW27 44405467 IC50 = 0.3 nM T10265 CR05OY 44405507 IC50 = 2.3 nM T10265 C7OA9V 44405510 IC50 = 0.3 nM T10265 CFY36C 44410864 IC50 = 1.2 nM T10265 CT1JW4 44410870 IC50 = 0.1 nM T10265 C3EI4T 44410882 IC50 = 40 nM T10265 C7NKA2 44410914 IC50 = 7000 nM T10265 CR0OV8 44441784 IC50 = 350 nM T10265 CBTQ53 44441786 IC50 = 670 nM T10265 C9Y2WJ 44441788 IC50 = 470 nM T10265 CL87OY 44441790 IC50 = 470 nM T10265 C1HK9B 44441792 IC50 = 390 nM T10265 CC06NP 44441794 IC50 = 310 nM T10265 C2AE1R 44441796 IC50 = 80 nM T10265 C4R7JV 44441798 IC50 = 88 nM T10265 C6DKS1 44441800 IC50 = 53 nM T10265 C1NZE3 44441802 IC50 = 24 nM T10265 C7FJE6 44441803 IC50 = 76 nM T10265 CU14PS 44441804 IC50 = 580 nM T10265 CGW2V9 44441813 IC50 = 110 nM T10265 C3JSH9 44441816 IC50 = 62 nM T10265 CSIA41 44441818 IC50 = 31 nM T10265 CR3JF0 44441820 IC50 = 17 nM T10265 CUH9C3 44441823 IC50 = 49 nM T10265 CM13IX 44441825 IC50 = 1.4 nM T10265 CSD1Q8 44441827 IC50 = 4.3 nM T10265 CG49SA 44441829 IC50 = 2 nM T10265 C8FK0V 44441831 IC50 = 1.6 nM T10265 CTI03C 44441833 IC50 = 1 nM T10265 CZYW49 44441837 IC50 = 2.2 nM T10265 CQ0N7Y 44441840 IC50 = 1.2 nM T10265 CENH10 44453381 IC50 = 4010 nM T10265 CY6XQ2 44453676 IC50 = 1090 nM T10265 CO3B2H 44453702 IC50 = 3070 nM T10265 CP7R6B 44453703 IC50 = 2870 nM T10265 C5PZF7 44453704 IC50 = 4130 nM T10265 CVY0F4 44453752 IC50 = 1850 nM T10265 CGK59A 44453754 IC50 = 30420 nM T10265 CH1JN6 44453755 IC50 = 1940 nM T10265 CY3HZ4 44453780 IC50 = 3080 nM T10265 CF73GI 44453781 IC50 = 890 nM T10265 C1KIE0 44476086 IC50 = 0.01 nM T10265 C48GWY 44518169 IC50 = 0.02512 nM T10265 CKI82C 44518336 IC50 = 0.03981 nM T10265 CSO35V 44520546 IC50 = 0.01585 nM T10265 C3HDX0 44561049 IC50 > 31622.78 nM T10265 CE2P6T 44561050 IC50 = 1995.26 nM T10265 CPQ14B 44561051 IC50 = 100 nM T10265 CE4T0V 44561052 IC50 = 50.12 nM T10265 CKQ8U6 44561053 IC50 = 12.59 nM T10265 C0LIF5 44561080 IC50 = 1000 nM T10265 C9A1GZ 44561081 IC50 = 316.23 nM T10265 C3V7MC 44561082 IC50 = 251.19 nM T10265 CIL03S 44561083 IC50 = 2511.89 nM T10265 CCW9Z4 44561084 IC50 = 199.53 nM T10265 C87UEF 44561085 IC50 = 3981.07 nM T10265 CS1U7C 44561086 IC50 = 5011.87 nM T10265 CN2QR1 44561087 IC50 = 158.49 nM T10265 CR58DF 44561088 IC50 = 3162.28 nM T10265 CS8X4Q 44561089 IC50 = 50.12 nM T10265 CEO2S3 44561090 IC50 = 125.89 nM T10265 CL58XP 44561091 IC50 = 100 nM T10265 C32KVC 44564728 IC50 = 100 nM T10265 C18OWC 44564729 IC50 > 31622.78 nM T10265 CHY5S7 44564730 IC50 > 31622.78 nM T10265 CX75RG 44564773 IC50 = 100 nM T10265 C28ESW 44564774 IC50 = 79.43 nM T10265 CA41KQ 44564808 IC50 = 5011.87 nM T10265 C9PB6G 44564809 IC50 = 6.31 nM T10265 C6H8QX 44564810 IC50 = 3162.28 nM T10265 C7Z8FW 44564811 IC50 = 19952.62 nM T10265 C7SK6C 44564844 IC50 = 1000 nM T10265 C97WTS 44564845 IC50 = 501.19 nM T10265 CLI0T3 44564846 IC50 = 251.19 nM T10265 CRF2P4 44564847 IC50 = 12589.25 nM T10265 C34WJG 44564894 IC50 = 3162.28 nM T10265 CV38ZJ 44564895 IC50 = 19952.62 nM T10265 CRKZ38 44564896 IC50 = 15848.93 nM T10265 CME04X 44564897 IC50 = 7943.28 nM T10265 CW8QC7 44564939 IC50 = 5.012 nM T10265 CJD73U 44565305 Ki = 500 nM T10265 CBL2J9 45263650 IC50 > 10000 nM T10265 CX5Q1U 45484316 IC50 = 5011.87 nM T10265 CO1NT8 45484317 IC50 = 5011.87 nM T10265 CG03XH 45484327 IC50 = 1258.93 nM T10265 CG1S6M 45484341 IC50 = 50.12 nM T10265 C19WRQ 45484346 IC50 = 100 nM T10265 CT53FB 45484347 IC50 = 398.11 nM T10265 CC20KO 45484400 IC50 > 10000 nM T10265 CY6NB1 45485421 IC50 = 12.59 nM T10265 C0CKG9 45485427 IC50 = 3.162 nM T10265 CUW0D1 45485428 IC50 = 199.53 nM T10265 C5BJS3 45485430 IC50 = 39.81 nM T10265 CJDP08 45485431 IC50 = 39.81 nM T10265 C3PD5Q 45485432 IC50 = 158.49 nM T10265 C4SQK9 45485433 IC50 = 0.631 nM T10265 CJCM05 45485435 IC50 = 0.01 nM T10265 CSVY10 45485439 IC50 = 1.585 nM T10265 C46RET 45485444 IC50 = 1.995 nM T10265 CFOS93 45485445 IC50 = 10 nM T10265 CP1TH3 45485455 IC50 = 6.31 nM T10265 CYQ3G8 45862748 IC50 = 68000 nM T10265 CMIE96 46213946 IC50 = 0.05 nM T10265 C2KE9Q 46227760 IC50 < 1 nM T10265 CN71UX 46227776 IC50 < 0.5012 nM T10265 CD8NU1 46238606 IC50 = 0.05 nM T10265 CO5J9W 46238636 IC50 = 0.03 nM T10265 CBU1I2 46238645 IC50 = 0.08 nM T10265 CPK53B 46238647 IC50 = 0.14 nM T10265 C92FLS 46238653 IC50 = 0.16 nM T10265 C48XRJ 46238655 IC50 = 4.83 nM T10265 C4XI0E 46238660 IC50 = 0.08 nM T10265 CES60L 46238684 IC50 = 0.014 nM T10265 C5H9JS 46238686 IC50 = 0.13 nM T10265 CXI4A9 46238694 IC50 = 0.085 nM T10265 C4MZ7W 46238696 IC50 = 0.38 nM T10265 C0I1XV 46238729 IC50 = 0.35 nM T10265 CD5ZQ1 46238730 IC50 = 0.06 nM T10265 CBI29N 46238731 IC50 = 0.35 nM T10265 C6CY8F 46238738 IC50 = 0.24 nM T10265 CL1U5W 46238739 IC50 = 0.04 nM T10265 C2CTG6 46238740 IC50 = 0.06 nM T10265 CFO26B 46238742 IC50 = 0.6 nM T10265 C5IMB2 46239424 Ki > 10000 nM T10265 CKR9P7 46239425 Ki > 10000 nM T10265 C3L9OR 46240228 IC50 = 0.03 nM T10265 CTX79H 46816028 IC50 = 41600 nM T10265 C1JOF3 46830337 Ki = 41 nM T10265 C3RJL6 46830338 Ki = 5.6 nM T10265 C7KW8T 46883839 IC50 = 19952.62 nM T10265 CZSG25 46883893 IC50 = 12589.25 nM T10265 C1YXQ7 46884033 Ki = 2600 nM T10265 CR75HO 46884094 Ki = 4300 nM T10265 C6TW3L 46884095 Ki = 1440 nM T10265 C7GJO6 46884096 Ki = 2010 nM T10265 C8DW2I 46884097 Ki = 2700 nM T10265 CGW26E 46884133 Ki = 1030 nM T10265 CZ2V3A 46884134 Ki = 210 nM T10265 C8HJV2 46884135 Ki = 1900 nM T10265 CE8SV7 46884136 Ki = 4900 nM T10265 CK7PD2 46884170 Ki = 14000 nM T10265 CR5AU2 46884171 Ki = 2700 nM T10265 CHBX41 46884172 Ki = 5200 nM T10265 C9B0QC 46884216 Ki = 413 nM T10265 CT1U9Q 46884217 Ki = 241 nM T10265 CSDA49 46884218 Ki = 26200 nM T10265 CZ9T7B 46884219 Ki = 5500 nM T10265 C35KWX 46884255 Ki = 4400 nM T10265 CW8EK3 46884256 Ki = 1000 nM T10265 C67OIK 46884257 Ki = 52200 nM T10265 CJ36UA 46884298 Ki = 432 nM T10265 CW1L6Q 46884299 Ki = 238 nM T10265 CHF10C 46884300 Ki = 5080 nM T10265 C8I2CM 46884366 Ki = 977 nM T10265 CVM1Q7 46884367 Ki = 222 nM T10265 CPT67V 46884368 Ki = 4440 nM T10265 C0L7JC 46884416 Ki = 77 nM T10265 CF0PI3 46915888 IC50 = 2.8 nM T10265 C3P2IN 46933992 IC50 = 45 nM T10265 CB2HS9 46933993 IC50 = 8.7 nM T10265 CZ7C3F 46933994 IC50 = 15.3 nM T10265 CPO7I1 49780545 IC50 = 333 nM T10265 CC7Q4R 49780546 IC50 = 865 nM T10265 CN7VO0 49780547 IC50 = 51 nM T10265 CQ5NF4 49780548 IC50 = 9.9 nM T10265 C9H4BC 49780549 IC50 = 40 nM T10265 C0EH7V 49865602 IC50 = 120 nM T10265 C89UPD 49865603 IC50 = 96.3 nM T10265 CV81PG 49865604 IC50 = 92.7 nM T10265 C43XGJ 49865605 IC50 = 43.3 nM T10265 CIT05Z 49865642 IC50 = 369 nM T10265 C5OI1V 49865643 IC50 = 57.6 nM T10265 C19JZB 49866243 IC50 = 10.7 nM T10265 CU5B8G 49866268 IC50 = 7.4 nM T10265 CSYL46 49866269 IC50 = 87 nM T10265 CI3F7K 49866270 IC50 = 389 nM T10265 C7V8DY 49866271 IC50 = 418 nM T10265 CCJ7I1 49866272 IC50 = 86.5 nM T10265 CN41YJ 50925469 IC50 > 50000 nM T10265 CQ3RG5 50925470 IC50 = 3600 nM T10265 CU8AL5 53244202 IC50 = 31000 nM T10265 C0OR7K 53248667 IC50 = 2580 nM T10265 C24HYO 53248668 IC50 = 2610 nM T10265 CS3R1I 53248669 IC50 = 120 nM T10265 C30RNE 53248670 IC50 = 55 nM T10265 CC5FO7 53346230 IC50 = 2.1 nM T10265 C6JR3L 53492818 IC50 = 0.17 nM T10265 CB85DI 53492819 IC50 = 1.2 nM T10265 C15PUI 53492820 IC50 = 0.43 nM T10265 COU3P7 53492821 IC50 = 0.75 nM T10265 CFCV89 53492822 IC50 = 13 nM T10265 CTZ20Y 53492823 IC50 = 2000 nM T10265 C7TMO3 53492943 IC50 = 0.32 nM T10265 CTQJ54 53492944 IC50 = 0.045 nM T10265 C46QKS 53492945 IC50 = 0.89 nM T10265 C9UOW4 53492946 IC50 = 0.27 nM T10265 CLV8Y3 53492947 IC50 = 0.11 nM T10265 CZ0Q2K 53493858 IC50 = 1.6 nM T10265 CW3A2S 53493859 IC50 = 12 nM T10265 CWU3P0 53493860 IC50 = 11 nM T10265 CI6EB9 53493990 IC50 = 3.3 nM T10265 C5RX6L 53493991 IC50 = 24 nM T10265 CW63RS 53493992 IC50 = 8.2 nM T10265 C3BYZ1 53493993 IC50 = 0.28 nM T10265 C8M6LN 53493994 IC50 = 0.35 nM T10265 C20EGY 53493995 IC50 = 0.23 nM T10265 CR0FY3 53494121 IC50 = 1.8 nM T10265 C92RJZ 53494122 IC50 = 8.4 nM T10265 CT5XR0 53494123 IC50 = 32 nM T10265 CX17GM 53494124 IC50 = 1.6 nM T10265 C6Z5RD 53494126 IC50 = 27 nM T10265 CM54WC 53494259 IC50 = 25 nM T10265 CWAX89 53494260 IC50 = 1.5 nM T10265 CR9B5K 53494261 IC50 = 2.3 nM T10265 CH1NR2 53494262 IC50 = 12 nM T10265 CK4T6M 53494263 IC50 = 12 nM T10265 C43JWF 53494264 IC50 = 3.6 nM T10265 CAM8R0 53494265 IC50 = 51 nM T10265 CRYH65 53494400 IC50 = 0.96 nM T10265 C9RNH7 53494402 IC50 = 120 nM T10265 CS5O1R 53494403 IC50 = 2400 nM T10265 C9BRW4 53494535 IC50 = 52 nM T10265 CU9H7X 53494536 IC50 = 8.5 nM T10265 C2WKM5 53494537 IC50 = 2.1 nM T10265 C12TDP 53494539 IC50 = 7.2 nM T10265 CG4AK1 53494665 IC50 = 14 nM T10265 C2UFG6 53494666 IC50 = 2.3 nM T10265 CU37MG 53494667 IC50 = 42 nM T10265 C5MWN0 53494668 IC50 = 5.6 nM T10265 CM01YV 53494669 IC50 = 5.6 nM T10265 CI9OD3 53494670 IC50 = 11 nM T10265 C7BV4A 53494798 IC50 = 9.6 nM T10265 CR4L7K 53494799 IC50 = 640 nM T10265 CMNU41 53494800 IC50 = 56 nM T10265 CQC3A6 53494801 IC50 = 0.89 nM T10265 C75QHZ 53494802 IC50 = 8.7 nM T10265 CX45GL 53494803 IC50 = 0.11 nM T10265 C9GXQ3 53495160 IC50 = 5 nM T10265 CC18WN 54579989 IC50 = 1300 nM T10265 CZM4S8 54579990 IC50 = 34 nM T10265 CDR9V3 54580135 IC50 = 940 nM T10265 C1RJ7M 54580520 IC50 > 400000 nM T10265 CCXF36 54580521 IC50 = 200000 nM T10265 CZG36N 54580522 IC50 = 11000 nM T10265 C0NPM8 54580523 IC50 = 17000 nM T10265 C25VSX 54580524 IC50 = 1700 nM T10265 C7A8SG 54580991 IC50 > 1000 nM T10265 CX1LD8 54581119 IC50 = 860 nM T10265 C9H8CS 54581120 IC50 = 150 nM T10265 C26WKU 54582010 IC50 = 57 nM T10265 C0MN3D 54582527 IC50 = 73000 nM T10265 C6T1QX 54582528 IC50 = 39000 nM T10265 CP4N1Q 54582529 IC50 = 2500 nM T10265 CHX67D 54582979 IC50 > 1000 nM T10265 C2RD7T 54583103 IC50 = 320 nM T10265 C3YD5S 54583104 IC50 = 78 nM T10265 CS0A2F 54583105 IC50 = 6.8 nM T10265 CW1X3G 54583497 IC50 > 400000 nM T10265 CP1ZD8 54583972 IC50 = 430 nM T10265 CJ5ZV7 54584101 IC50 = 1200 nM T10265 CQPH74 54584479 IC50 = 1380 nM T10265 CF3HA7 54585042 IC50 = 120 nM T10265 C3-FEB-08 54585043 IC50 = 2800 nM T10265 CG54MF 54585044 IC50 = 190 nM T10265 CN96IQ 54585432 IC50 = 115000 nM T10265 CAI3B7 54585882 IC50 = 140 nM T10265 CBF2W8 54586013 IC50 = 690 nM T10265 CYI6K8 54586014 IC50 = 1800 nM T10265 C38ZLC 54586015 IC50 = 600 nM T10265 CH25CO 54586393 IC50 = 16000 nM T10265 C82LED 54586394 IC50 = 2000 nM T10265 CT1A3P 54586846 IC50 = 120 nM T10265 CY6QC5 54586847 IC50 > 1000 nM T10265 CK6QW0 54586848 IC50 = 300 nM T10265 C2FN8X 54586849 IC50 = 540 nM T10265 COU0I7 54586989 IC50 > 1000 nM T10265 C8IO0C 54586990 IC50 = 3700 nM T10265 C3L9NI 54586991 IC50 = 220 nM T10265 C52NHY 54586992 IC50 = 210 nM T10265 C5DO4H 54586993 IC50 = 220 nM T10265 CXR9T5 54586994 IC50 = 34 nM T10265 CQ1H3C 54587403 IC50 = 30000 nM T10265 C28GAC 54587404 IC50 = 16000 nM T10265 C43HNS 54588470 IC50 = 2.7 nM T10265 C04EUG 56589630 IC50 = 0.02 nM T10265 CHT86A 56642417 IC50 = 8.7 nM T10265 CBV60W 56642529 IC50 = 0.8 nM T10265 CKGD94 56642530 IC50 = 24 nM T10265 CKTD52 56642531 IC50 = 2.1 nM T10265 C4G6TL 56642532 IC50 = 19 nM T10265 CRK35Q 56642533 IC50 = 1.7 nM T10265 CF7P1Y 56642534 IC50 = 25 nM T10265 CP9CD7 56642658 IC50 = 9.7 nM T10265 CM8U9E 56642659 IC50 = 4.3 nM T10265 CAN50G 56642660 IC50 = 0.2 nM T10265 C1AND4 56659469 IC50 = 17 nM T10265 CGWH19 56662928 IC50 = 32 nM T10265 CQT17K 56662929 IC50 = 0.51 nM T10265 CLMG01 56662930 IC50 = 0.52 nM T10265 CL1U3W 56666405 IC50 = 0.66 nM T10265 C5H9XA 56669821 IC50 = 0.55 nM T10265 CIX9M0 56673307 IC50 = 0.46 nM T10265 CTY48D 56673902 IC50 = 4.6 nM T10265 CEO42M 56676640 IC50 = 0.58 nM T10265 C2CRW3 56679969 IC50 = 1 nM T10265 CT8A6K 56683302 IC50 = 0.35 nM T10265 C6RD5I 56834321 IC50 = 5600 nM T10265 C29UZH 56834322 IC50 = 75800 nM T10265 CJ9XQ5 56834424 IC50 = 16800 nM T10265 CT60PE 56834425 IC50 = 68100 nM T10265 CWZ0Y6 56834426 IC50 = 29400 nM T10265 CLU7B8 56834427 IC50 = 65100 nM T10265 CSW83T 56834428 IC50 = 20100 nM T10265 CZJ53R 56834429 IC50 = 10200 nM T10265 CBGS50 56834430 IC50 = 6400 nM T10265 CKG24D 56834431 IC50 = 21700 nM T10265 CF76QM 56834432 IC50 = 78100 nM T10265 CS79EV 56834529 IC50 = 18700 nM T10265 CEM95R 56834530 IC50 = 2800 nM T10265 C9U7JL 56834531 IC50 = 3900 nM T10265 CUCZ73 56834532 IC50 = 56800 nM T10265 CSA47G 56834533 IC50 = 47800 nM T10265 CCS31I 56834534 IC50 = 20700 nM T10265 CZR27O 56834535 IC50 = 27900 nM T10265 CWX80D 56834536 IC50 = 8700 nM T10265 CLB1Q6 56834537 IC50 = 4800 nM T10265 CW7KJ4 56834625 IC50 = 36700 nM T10265 C6WD4G 56834626 IC50 = 65700 nM T10265 CAP53L 56834627 IC50 = 5600 nM T10265 CL4U1G 56834628 IC50 = 1200 nM T10265 C3ZRD5 56929886 IC50 = 1520 nM T10265 C0ZF1L 57328385 IC50 = 7000 nM T10265 CBR49P 57334265 IC50 = 265 nM T10265 C2G9PX 57345604 IC50 = 350 nM T10265 C2BND3 57384028 EC50 = 890 nM T10265 CB17SC 57385767 IC50 = 12400 nM T10265 CD52CA 57391118 IC50 > 2000 nM T10265 CG3DF1 57392948 Ki > 10000 nM T10265 CE36TV 57394695 Ki > 10000 nM T10265 CB21SH 57398742 IC50 = 380 nM T10265 C7VMN0 57398767 IC50 = 260 nM T10265 CD5W3L 57399439 IC50 = 284 nM T10265 C5BM4F 57400402 IC50 = 3490 nM T10265 CTO39H 57401200 IC50 = 280 nM T10265 C36SZR 57401201 IC50 = 278 nM T10265 CZ81YC 57401202 IC50 = 257 nM T10265 CS8LW0 57401203 IC50 = 251 nM T10265 CPA3D1 57403394 Ki > 10000 nM T10265 CDA74Z 57600658 IC50 = 1.2 nM T10265 C6FY8M 57600737 IC50 = 0.3 nM T10265 CR6Z9C 57600809 IC50 = 0.7 nM T10265 C2PGE3 57600813 IC50 = 0.03 nM T10265 CLK8O5 57600820 IC50 = 3.7 nM T10265 C36WCS 57600842 IC50 = 0.81 nM T10265 C3EM8A 57600926 IC50 = 26 nM T10265 C7O5HY 57600960 IC50 = 0.3 nM T10265 CK7L8X 57601096 IC50 = 4.3 nM T10265 CN8D4I 57601175 IC50 = 0.1 nM T10265 CU61GM 57601298 IC50 = 0.36 nM T10265 C0PXR1 57601304 IC50 = 0.05 nM T10265 CNH5Y7 57601312 IC50 = 1.8 nM T10265 C81JFC 57601337 IC50 = 0.46 nM T10265 C78XOS 57601386 IC50 = 37 nM T10265 C6LY3S 57601465 IC50 = 1.5 nM T10265 CYM0K3 57601557 IC50 = 3.4 nM T10265 C2IPY1 57601592 IC50 = 0.5 nM T10265 CNP13J 57601655 IC50 = 1.6 nM T10265 CVB98S 57601701 IC50 = 0.35 nM T10265 C4PAR9 57601713 IC50 = 0.11 nM T10265 CD5CJ9 57601760 IC50 = 2.7 nM T10265 CL3EN6 57601817 IC50 = 4.1 nM T10265 C1HF7E 57601851 IC50 = 0.04 nM T10265 C57LTR 57602000 IC50 = 0.7 nM T10265 C6XR8W 57602004 IC50 = 0.9 nM T10265 CLBQ42 57602014 IC50 = 12.7 nM T10265 CA4IZ2 58013972 IC50 = 39 nM T10265 CYJ53N 58014021 IC50 = 750 nM T10265 C8N0QY 59190402 IC50 = 0.03162 nM T10265 CNXQ37 59190421 IC50 = 0.03162 nM T10265 C5WT7D 59190424 IC50 = 0.05012 nM T10265 C60AHZ 59190427 IC50 = 0.05012 nM T10265 C50KJN 59190428 IC50 = 0.03162 nM T10265 C1BE3Q 59190429 IC50 = 0.01995 nM T10265 C6D3JY 59190434 IC50 = 0.07943 nM T10265 CR59YI 59190438 IC50 = 0.01585 nM T10265 CZD16C 59190442 IC50 = 0.01995 nM T10265 COFA01 59190446 IC50 = 0.01995 nM T10265 C19AUN 59190447 IC50 = 0.05012 nM T10265 CW24YS 59190451 IC50 = 0.01995 nM T10265 CQ1SG7 59190453 IC50 = 0.1 nM T10265 CKG2Z8 59190459 IC50 = 0.03162 nM T10265 C3TEH1 59190462 IC50 = 0.01585 nM T10265 C6DG2S 59190464 IC50 = 0.03981 nM T10265 CU3YL9 59190469 IC50 = 0.1 nM T10265 CT40JG 59190479 IC50 = 0.0631 nM T10265 C4GBR3 59190483 IC50 = 0.03162 nM T10265 CE0HQ8 59190485 IC50 = 0.0631 nM T10265 CF8JG6 59190501 IC50 = 0.07943 nM T10265 CL9R5M 59190503 IC50 = 0.0631 nM T10265 C7P6QI 59190515 IC50 = 0.01995 nM T10265 CYI46M 59190526 IC50 = 0.7943 nM T10265 C0Q8XF 59190527 IC50 = 0.3981 nM T10265 C5R1FQ 59190528 IC50 = 0.02512 nM T10265 CEI8A5 59190544 IC50 = 0.02512 nM T10265 CQHS47 59190547 IC50 = 0.02512 nM T10265 C79GHB 59190548 IC50 = 0.01995 nM T10265 C2UMO9 59190556 IC50 = 0.1259 nM T10265 C2XDK5 59190565 IC50 = 0.1259 nM T10265 C7GW8Y 59227395 IC50 = 2.7 nM T10265 CQ32HT 59227396 IC50 = 0.27 nM T10265 C54GSB 59227397 IC50 = 0.19 nM T10265 CLG2T6 59227400 IC50 = 550 nM T10265 C09PJC 59227401 IC50 = 1.5 nM T10265 C0EQ5D 59227405 IC50 = 9.8 nM T10265 CZI9U7 59227406 IC50 = 2.9 nM T10265 COJ94S 59227408 IC50 = 9.4 nM T10265 CSC67X 59227409 IC50 = 21 nM T10265 C9C8TZ 59227411 IC50 = 4.5 nM T10265 C34SNK 59227413 IC50 = 0.11 nM T10265 CVH8T2 59227421 IC50 = 39 nM T10265 C1BU7R 59227423 IC50 = 83 nM T10265 COC80E 59335994 IC50 = 0.77 nM T10265 CN62MK 59336034 IC50 = 2580 nM T10265 CB9GO8 59336035 IC50 = 3.2 nM T10265 CF0Q4T 60150541 IC50 = 4570 nM T10265 CW37UH 67548131 IC50 = 0.05 nM T10265 C56UIN 67548175 IC50 = 0.05 nM T10265 C6VKP4 67548337 IC50 = 0.05 nM T10265 C9JLW2 67548347 IC50 = 0.7 nM T10265 CGXY26 67548392 IC50 = 0.03 nM T10265 C5U3WL 67548498 IC50 = 0.05 nM T10265 C6LA7R 67548508 IC50 = 0.05 nM T10265 CC4Y6V 67548720 IC50 = 0.04 nM T10265 C8B1JS 67548983 IC50 = 0.37 nM T10265 CPQ2I7 67549056 IC50 = 0.09 nM T10265 C71HZU 67549086 IC50 = 0.05 nM T10265 C74YXW 67549097 IC50 = 0.21 nM T10265 CD09WI 67549451 IC50 = 0.31 nM T10265 C5M0NT 67549626 IC50 = 0.22 nM T10265 C05LWV 67549660 IC50 = 0.11 nM T10265 C8Z7RX 67549879 IC50 = 0.06 nM T10265 C18CNK 68405754 IC50 = 0.03 nM T10265 CNYS04 68405874 IC50 = 0.15 nM T10265 CWEQ54 68405927 IC50 = 0.03 nM T10265 CM4WP6 68406148 IC50 = 1.7 nM T10265 C4ZEH9 68578314 IC50 = 2560 nM T10265 C8H4JX 70681173 IC50 = 50.12 nM T10265 C2Y8DO 70685261 IC50 = 8.4 nM T10265 CK7Y2D 70686701 IC50 = 3.4 nM T10265 COM2C3 70690671 IC50 = 480 nM T10265 C4P0XT 71092344 IC50 = 0.0278 nM T10265 C6DAG4 71092519 IC50 = 0.0881 nM T10265 C0O6TB 71254628 IC50 = 4.7 nM T10265 CWF39E 71254723 IC50 = 910 nM T10265 C93LAB 71254931 IC50 = 4 nM T10265 CF90QO 71262535 IC50 = 180 nM T10265 C14TJO 71262536 IC50 = 740 nM T10265 C7AQH0 71262640 IC50 = 1.8 nM T10265 CU7DZ1 71262641 IC50 = 5.4 nM T10265 C7LRS9 71305062 IC50 = 378 nM T10265 CJ62MK 71451776 IC50 = 47 nM T10265 C2UK6B 71451779 IC50 = 53 nM T10265 CJ3Z7K 71460703 IC50 = 4.6 nM T10265 CJS9R6 71463568 IC50 = 11 nM T10265 CHD9Q2 71512292 IC50 = 21 nM T10265 C13OKG 71517744 IC50 = 0.66 nM T10265 C54EWN 71517745 IC50 = 0.3 nM T10265 CKOZ85 71517907 IC50 = 5.9 nM T10265 CB0OK6 71517908 IC50 = 6 nM T10265 CC8GZ6 71517909 IC50 = 0.1 nM T10265 CP9G6K 71517910 IC50 = 20 nM T10265 CP6DN1 71517911 IC50 = 0.5 nM T10265 C6D7EY 71518079 IC50 = 0.064 nM T10265 C83PUL 71518080 IC50 = 1.4 nM T10265 CBJZ01 71518081 IC50 = 0.3 nM T10265 C7Q2GV 71518082 IC50 = 3.1 nM T10265 C40KMI 71518243 IC50 = 2.7 nM T10265 CJ36SE 71518244 IC50 = 20 nM T10265 CNZ3L1 71552789 IC50 = 540 nM T10265 CYZS90 71552873 IC50 = 1570 nM T10265 C3MOC4 71562032 IC50 = 1093 nM T10265 C5XT1F 71562033 IC50 = 601 nM T10265 CCO9D5 71562034 IC50 = 394 nM T10265 CM71TP 71562154 IC50 = 235 nM T10265 CQBC15 71562381 IC50 = 282 nM T10265 C4YM5X 71562382 IC50 = 278 nM T10265 C51KEM 71562383 IC50 = 271 nM T10265 C3HV9Y 71562696 IC50 = 1100 nM T10265 CTJ1N2 71583536 IC50 = 1230 nM T10265 C28DSF 71583538 IC50 = 530 nM T10265 C4GNJ3 71598545 IC50 = 0.87 nM T10265 C2YCS7 71624531 IC50 = 583 nM T10265 CZ4KC3 71624641 IC50 = 1950 nM T10265 CUWS89 71624642 IC50 = 330 nM T10265 C5NU1X 71624751 IC50 = 100000 nM T10265 CPBJ05 71624752 IC50 = 100000 nM T10265 CFD0X9 71624753 IC50 = 8160 nM T10265 CMQ7N9 71624754 IC50 = 2070 nM T10265 C4FC1W 71624755 IC50 = 8110 nM T10265 C9D5MC 71624843 IC50 = 150 nM T10265 C02RYV 71624844 IC50 = 610 nM T10265 CUB7Z0 71624845 IC50 = 430 nM T10265 CO7X9M 71624869 IC50 = 100000 nM T10265 C3OTL4 71624870 IC50 = 27000 nM T10265 C4WN1T 71624871 IC50 = 6190 nM T10265 C2UZC5 71624872 IC50 = 6740 nM T10265 CZF6X3 71624873 IC50 = 5660 nM T10265 CFCD52 71624959 IC50 = 2200 nM T10265 CZF36U 71624960 IC50 = 480 nM T10265 CXFZ54 71624962 IC50 = 230 nM T10265 C0WZ3P 71624963 IC50 = 29 nM T10265 C6SP8E 71624964 IC50 = 25 nM T10265 COUW49 71624965 IC50 = 28 nM T10265 CBX7F6 71624993 IC50 = 1920 nM T10265 CJ1K6H 71624994 IC50 = 110 nM T10265 CG9ZJ8 71624995 IC50 = 534 nM T10265 CFL69D 71624996 IC50 = 741 nM T10265 CV69IU 71624997 IC50 = 138 nM T10265 CY54HG 71625090 IC50 = 280 nM T10265 CW71GU 71625091 IC50 = 7900 nM T10265 C8ANX9 71625092 IC50 = 16 nM T10265 C6NW7K 71625095 IC50 = 29 nM T10265 C16JZP 71625120 IC50 = 410 nM T10265 C5CQM8 71625121 IC50 = 265 nM T10265 C7XL9G 71625122 IC50 = 418 nM T10265 C2N1FS 71625123 IC50 = 695 nM T10265 C61ULV 71625124 IC50 = 353 nM T10265 CF72LN 71625226 IC50 = 190 nM T10265 CG2BF3 71625227 IC50 = 5000 nM T10265 C98AKE 71625228 IC50 = 3000 nM T10265 CJO96Q 71625229 IC50 = 140 nM T10265 C7M9TR 71625230 IC50 = 2500 nM T10265 C0C1GB 71625231 IC50 = 800 nM T10265 C7Z5GP 71625256 IC50 = 562 nM T10265 C5GQ7K 71625349 IC50 = 27 nM T10265 C1TNV3 71625350 IC50 = 7.5 nM T10265 C3HMB0 71625351 IC50 = 70 nM T10265 CB0MK4 71625352 IC50 = 6.6 nM T10265 C7A3ZT 71625461 IC50 = 4.7 nM T10265 C59HQL 71625462 IC50 = 43 nM T10265 C32MVE 71625463 IC50 = 33 nM T10265 CVFT59 71653160 IC50 > 5000 nM T10265 CY1P2J 71657973 IC50 = 17000 nM T10265 C68SDB 71719394 IC50 = 0.5012 nM T10265 CUJ15C 71719800 IC50 = 4220 nM T10265 CK1WI4 71741428 IC50 = 8.3 nM T10265 CT4RA0 72188901 IC50 = 50 nM T10265 CT3L6W 72188902 IC50 = 22 nM T10265 CGJR02 72192867 IC50 = 240 nM T10265 C38UIK 72192868 IC50 = 150 nM T10265 CU43LO 72193176 IC50 = 1260 nM T10265 CQI8K4 72193177 IC50 = 980 nM T10265 C9ONF0 72193178 IC50 = 10200 nM T10265 C5KPN6 72193179 IC50 = 570 nM T10265 C4MKD5 72193180 IC50 = 6130 nM T10265 CF3Y7X 72193181 IC50 = 16600 nM T10265 CBL5P7 72697147 IC50 = 200 nM T10265 C5SQ8X 72697148 IC50 = 4000 nM T10265 CFRO57 72697149 IC50 = 2000 nM T10265 C6YGJ9 72697150 IC50 = 47 nM T10265 C4K5ZS 72697151 IC50 = 7.3 nM T10265 CF4TM9 72697287 IC50 = 8200 nM T10265 CBV2E0 72697290 IC50 = 120 nM T10265 CY87JM 72697291 IC50 = 120 nM T10265 CJ02FY 72697292 IC50 = 16 nM T10265 CMF48I 72697293 IC50 = 11 nM T10265 COH2F6 72697436 IC50 = 110 nM T10265 CD6Q1P 72697437 IC50 = 7.1 nM T10265 CPTM83 72697438 IC50 = 490 nM T10265 C01TZI 72697439 IC50 = 29 nM T10265 CNG3B5 72697440 IC50 = 110 nM T10265 CM0H9P 72697584 IC50 = 11 nM T10265 CA1GS3 72697585 IC50 = 8.2 nM T10265 C2YS6M 72697586 IC50 = 3.7 nM T10265 CK5O3E 72697587 IC50 = 16 nM T10265 CTL51Z 72697588 IC50 = 13 nM T10265 CJ81XO 72697727 IC50 = 6500 nM T10265 CO7YV4 72725405 IC50 = 4920 nM T10265 C08HDR 72947900 IC50 = 117 nM T10265 CVR10K 72947901 IC50 = 118 nM T10265 CPE27J 72947902 IC50 = 104 nM T10265 C3UH7M 72948092 IC50 = 92 nM T10265 CD3BZ0 73603954 IC50 = 220 nM T10265 CZ14AK 74220843 IC50 = 1642 nM T10265 CYB9G4 74220906 IC50 = 136 nM T10265 CXSH27 74220907 IC50 = 562 nM T10265 CLR80D 74221042 IC50 = 1945 nM T10265 CCZ1V0 74221043 IC50 = 8815 nM T10265 C7Y2JO 74221099 IC50 = 383 nM T10265 CBM14E 74221100 IC50 = 1394 nM T10265 CQ2KG4 74221101 IC50 = 261 nM T10265 CQGT60 74221102 IC50 = 4048 nM T10265 CL0P7R 74221104 IC50 = 2447 nM T10265 C8D4KG 74221105 IC50 = 251 nM T10265 CC37TX 74221165 IC50 = 237 nM T10265 C64ZJD 74221166 IC50 = 3770 nM T10265 CUTB06 74221167 IC50 = 135 nM T10265 C7IYQ1 74221168 IC50 = 781 nM T10265 CSP7M5 74221169 IC50 = 241 nM T10265 C3CSM1 74221170 IC50 = 1862 nM T10265 CLG7T8 74221229 IC50 = 46 nM T10265 CAUC08 74221233 IC50 = 1437 nM T10265 CB9GN2 74221235 IC50 = 135 nM T10265 C1QRG0 74221297 IC50 = 165 nM T10265 C6V1FJ 74221298 IC50 = 12 nM T10265 CX5H8N 74221299 IC50 = 126 nM T10265 CTU9V5 74221300 IC50 = 69 nM T10265 CH7K9G 74221301 IC50 = 24 nM T10265 C9WHR4 74221360 IC50 = 48 nM T10265 C04QOM 74221361 IC50 = 1090 nM T10265 CKBM41 74221363 IC50 = 1574 nM T10265 CPYO61 74221364 IC50 = 44 nM T10265 C15QVF 74221424 IC50 = 225 nM T10265 CDRO05 74221427 IC50 = 584 nM T10265 CB4M7E 74221497 IC50 = 105 nM T10265 CSXY74 74221498 IC50 = 11 nM T10265 C1LCQ5 76310584 IC50 = 13 nM T10265 CNY85L 76310585 IC50 = 30 nM T10265 CGN2F0 76310586 IC50 = 14 nM T10265 CS4GB6 76310587 IC50 = 3 nM T10265 CZWC27 76314221 IC50 = 120 nM T10265 CLXO82 76314222 IC50 = 140 nM T10265 CHKB59 76314223 IC50 = 38 nM T10265 CHC31S 76314224 IC50 = 250 nM T10265 CYC23W 76314225 IC50 = 10 nM T10265 C1X5GR 76314226 IC50 = 64 nM T10265 CDWE89 76317790 IC50 = 120 nM T10265 CFQ0P3 76317791 IC50 = 120 nM T10265 CPBL42 76317792 IC50 = 140 nM T10265 CWB80L 76317793 IC50 = 8.3 nM T10265 C4KH2T 76321500 IC50 = 880 nM T10265 C1XTZ7 76321501 IC50 = 10 nM T10265 C34RGJ 76321502 IC50 = 20 nM T10265 C1TS0Y 76321503 IC50 = 5.2 nM T10265 C93VYC 76321504 IC50 = 9.9 nM T10265 CENO19 76321505 IC50 = 3.8 nM T10265 C78QEP 76325104 IC50 = 57 nM T10265 CSMV71 76325105 IC50 = 11 nM T10265 CNBJ29 76325106 IC50 = 46 nM T10265 C5P9TA 76325107 IC50 = 4.6 nM T10265 CO8J5I 76328668 IC50 = 34 nM T10265 CP1T2G 76328669 IC50 = 71 nM T10265 CH5Z2P 76328670 IC50 = 19 nM T10265 CWM15I 76328671 IC50 = 7.5 nM T10265 CFA85S 76328672 IC50 = 5.9 nM T10265 C1A4WZ 76332343 IC50 = 78 nM T10265 C6R2XP 76332344 IC50 = 30 nM T10265 CW4Y7O 76332345 IC50 = 38 nM T10265 C2J6IZ 76332346 IC50 = 140 nM T10265 CTXG71 76332347 IC50 = 44 nM T10265 CCFA47 76332348 IC50 = 56 nM T10265 CWKO07 76335973 IC50 = 38 nM T10265 CL3D1Y 76335974 IC50 = 16 nM T10265 CB64TA 76335975 IC50 = 49 nM T10265 CXA0Y3 76335976 IC50 = 8.2 nM T10265 CY34OK 86280445 IC50 = 5900 nM T10265 C2AM7F 90110094 IC50 = 57 nM T10265 CEW76O 90110531 IC50 = 166 nM T10265 CTIC43 90111581 IC50 = 953 nM T10265 CF8I0P 90111742 IC50 = 43 nM T10265 CW7R5J 90112663 IC50 = 128 nM T10265 CNC5U2 90112840 IC50 = 58 nM T10265 C8BO3W 90113029 IC50 = 18755 nM T10265 C6EC4P 90113094 IC50 = 3830 nM T10265 CL1ZU8 90338511 IC50 = 1287 nM T10265 CLC17A 90338526 IC50 = 356 nM T10265 CSU1W0 90338537 IC50 = 1419 nM T10265 C2M8OK 90338579 IC50 = 137 nM T10265 CN1Q6Y 90643907 IC50 = 0.02512 nM T10265 CY8G2C 90643908 IC50 = 0.03162 nM T10265 CKD07U 90643909 IC50 = 0.3162 nM T10265 CC8S1P 90643910 IC50 = 2.512 nM T10265 CE9AH0 90643911 IC50 = 0.05012 nM T10265 C48ZJP 90643912 IC50 = 0.3162 nM T10265 C23UJE 90643913 IC50 = 19.95 nM T10265 CH0SA3 90643914 IC50 = 0.03162 nM T10265 CX46KU 90643915 IC50 = 0.1259 nM T10265 CRJ8D4 90665374 IC50 = 3430 nM T10265 C4RN9B 90667924 IC50 = 1330 nM T10265 CG5HV8 90668361 IC50 = 31500 nM T10265 C2HQ7I 90668362 IC50 = 5060 nM T10265 CDB74T 90668364 IC50 = 7100 nM T10265 C4BD5F 91667427 IC50 = 520 nM T10265 C45QVJ 91668196 IC50 = 46 nM T10265 C19SMQ 101133935 IC50 = 1.585 nM T10265 C2A7OZ 101133941 IC50 = 0.3162 nM T10265 C7ZRA5 101133943 IC50 = 0.1995 nM T10265 CQCA74 101886683 IC50 = 4400 nM T10265 C4LQ7R 101891513 IC50 = 380 nM T10265 C1T7MA 118037253 IC50 = 3287 nM T10265 C90MKD 118037440 IC50 = 98 nM T10265 C21HKZ 118048422 IC50 = 402 nM T10265 CW7TU1 118708069 IC50 = 1460 nM T10265 C2D0NW 118708070 IC50 = 2777 nM T10265 CE59WQ 118708071 IC50 = 2282 nM T10265 C6VT7X 118708072 IC50 = 845 nM T10265 CE1J8A 118710544 IC50 = 38 nM T10265 C2S9TF 118711358 IC50 = 18000 nM T10265 CR75BH 118712216 IC50 = 12 nM T10265 CJIY54 118712217 IC50 = 11 nM T10265 C0NQ6I 118712218 IC50 = 1700 nM T10265 C3XM4A 118712219 IC50 = 2700 nM T10265 C6KRJ9 118712220 IC50 = 5.5 nM T10265 C86PHO 118712221 IC50 = 8.8 nM T10265 CD82CM 118712222 IC50 = 88 nM T10265 C9NCB0 118719988 IC50 = 4900 nM T10265 CC4IU3 118719991 IC50 = 3500 nM T10265 CC48FZ 118719992 IC50 = 920 nM T10265 CX92KJ 118719994 IC50 = 3800 nM T10265 COLJ03 118719995 IC50 = 3700 nM T10265 C0Z3GQ 118719996 IC50 = 3000 nM T10265 CY2NS6 118719997 IC50 = 3200 nM T10265 C1WC8D 118719998 IC50 = 1400 nM T10265 C1UBR0 118719999 IC50 = 820 nM T10265 CB29OG 118720000 IC50 = 1100 nM T10265 CM6ZP8 118720001 IC50 = 3400 nM T10265 C8HP5T 118720002 IC50 = 720 nM T10265 CSIF10 118720003 IC50 = 3800 nM T10265 C1WE3G 118720004 IC50 = 480 nM T10265 CZYT12 118720005 IC50 = 1000 nM T10265 CW41JN 118720006 IC50 = 640 nM T10265 CU56DJ 118720007 IC50 = 520 nM T10265 CD6U4P 118720008 IC50 = 3300 nM T10265 C9U6TB 118724077 IC50 = 7400 nM T10265 CUQ6W2 118724078 IC50 = 4300 nM T10265 CP0X8J 118724083 IC50 = 2700 nM T10265 CWRL26 118724084 IC50 = 3000 nM T10265 C5B7AW 118724086 IC50 = 30000 nM T10265 CNM6F3 118724087 IC50 = 5300 nM T10265 CH4L6O 118724088 IC50 = 670 nM T10265 CCZ6W9 118724089 IC50 = 610 nM T10265 C40AXS 118724090 IC50 = 56 nM T10265 CKG08X 118724091 IC50 = 180 nM T10265 C3OR6T 118724092 IC50 = 310 nM T10265 CM6XW1 118724093 IC50 = 280 nM T10265 C46LFG 118724094 IC50 = 180 nM T10265 CYM21X 118724095 IC50 = 20 nM T10265 C5TL8H 118725359 IC50 = 30600 nM T10265 CE49ML 118725368 IC50 = 25900 nM T10265 CM8EO1 118729736 IC50 = 11000 nM T10265 CDHC56 118729740 IC50 = 4800 nM T10265 CEKR01 118729741 IC50 = 12000 nM T10265 CBJ24Z 118729742 IC50 = 24000 nM T10265 CL23ZS 118729745 IC50 = 550 nM T10265 CUW3D1 118729746 IC50 = 200 nM T10265 C1UL3B 118729747 IC50 = 420 nM T10265 C72ATF 118729748 IC50 = 1100 nM T10265 C59LGI 118729749 IC50 = 14000 nM T10265 CPQN92 118729750 IC50 = 25000 nM T10265 C5MI9E 118729751 IC50 = 440 nM T10265 CE5ON1 118729752 IC50 = 1500 nM T10265 CX0W4F 118729753 IC50 = 560 nM T10265 CB1DX3 118729754 IC50 = 1900 nM T10265 CC41IT 118729755 IC50 = 1400 nM T10265 CB2DX0 118729756 IC50 = 2300 nM T10265 CB40SN 118729757 IC50 = 380 nM T10265 C4HI1Q 118729758 IC50 = 200 nM T10265 CKBG19 118729759 IC50 = 140 nM T10265 CIL5N0 122190063 IC50 = 23500 nM T10265 COXC98 122190064 IC50 = 23300 nM T10265 CW1O4E 122190065 IC50 = 15500 nM T10265 CL6BG2 122190066 IC50 = 37000 nM T10265 CEX3R1 122190067 IC50 = 2300 nM T10265 COF4R0 122190068 IC50 = 43000 nM T10265 CT5KD1 122190069 IC50 = 26800 nM T10265 C6O4CS 122190070 IC50 = 37900 nM T10265 C26KOP 122190071 IC50 = 15700 nM T10265 CP2IA1 122190072 IC50 = 38100 nM T10265 CN6OD7 122190073 IC50 > 50000 nM T10265 CNR16E 122190074 IC50 > 50000 nM T10265 CS80MH 122193673 IC50 = 1031 nM T10265 C8CJU5 122193675 IC50 = 1087 nM T10265 CS6M9C 122193679 IC50 = 976 nM T10265 CJKO62 122193703 IC50 = 6420 nM T10265 C9W1JO 122193704 IC50 = 3800 nM T10265 C2MNX0 122193705 IC50 = 380 nM T10265 C5EHB7 122193706 IC50 = 1770 nM T10265 C5WI6U 122193707 IC50 = 1770 nM T10265 COT0R6 122193708 IC50 = 900 nM T10265 CJF36H 122193709 IC50 = 1580 nM T10265 C0J6MS 122193710 IC50 = 10300 nM T10265 C0XLR7 122193711 IC50 = 4800 nM T10265 CC9I0U 122193712 IC50 = 18300 nM T10265 CX30HD 122193713 IC50 = 1040 nM T10265 CQV4W1 122193754 IC50 = 301 nM T10265 C6IJH8 122193928 IC50 = 1020 nM T10265 CNT17O 122193929 IC50 = 4240 nM T10265 C6Q5UO 122193930 IC50 = 11600 nM T10265 C1SWM0 122193931 IC50 = 7310 nM T10265 C9JSX0 122193932 IC50 = 1730 nM T10265 C6GI3B 122193933 IC50 = 1590 nM T10265 C9PTW4 122193934 IC50 = 900 nM T10265 C5FKM8 122193935 IC50 = 760 nM T10265 CER6C8 127025905 IC50 = 0.5012 nM T10265 C7RL8G 127025906 IC50 = 0.631 nM T10265 CL8ZE4 127037893 IC50 = 1950 nM T10265 C2A3TY 127038253 IC50 = 38 nM T10265 C86UVX 127038665 IC50 = 26 nM T10265 CUA14O 127038666 IC50 = 7 nM T10265 CY2JI6 127039005 IC50 = 4 nM T10265 C3LWF7 127039006 IC50 = 7 nM T10265 CTLJ59 127039007 IC50 = 0.7 nM T10265 C8WQ5K 127039011 IC50 = 0.2 nM T10265 CSY34W 127039587 IC50 = 165 nM T10265 CW59OX 127039663 IC50 = 5 nM T10265 CQD37E 127040004 IC50 = 6 nM T10265 C8QM7X 127040005 IC50 = 0.2 nM T10265 CC71SR 127040006 IC50 = 0.1 nM T10265 C7V8RC 127040007 IC50 = 0.03 nM T10265 CI6J9N 127041241 IC50 > 10000 nM T10265 CCNA62 127041543 IC50 = 16 nM T10265 CW2HR1 130366728 IC50 = 6.51 nM T10265 C2ALN7 130366739 IC50 = 27.6 nM T10265 CQJN83 130366758 IC50 = 211 nM T10265 CDAF16 130380472 IC50 = 178 nM T10265 C18KLO 130380505 IC50 = 207 nM T10265 C5XCO1 130380512 IC50 = 26.7 nM T10265 CT2E8Q 130380575 IC50 = 55.6 nM T10265 CH0QB7 132471725 Ki = 3162.28 nM T10265 CQ1Y0K 132471729 Ki = 1995.26 nM T10265 CG8HF1 132938287 IC50 = 1600 nM T10265 C2P1IU 134129996 IC50 = 144 nM T10265 CLE03O 134130328 IC50 = 39 nM T10265 CSN6J0 134130563 IC50 = 34 nM T10265 C0A1CZ 134131162 IC50 = 166 nM T10265 CF3WB2 134131879 IC50 = 13080 nM T10265 CH9QG2 134132752 IC50 = 170 nM T10265 C83IYJ 134133852 IC50 = 1130 nM T10265 CYXE80 134133962 IC50 = 1410 nM T10265 C4UMZ5 134136652 IC50 = 1220 nM T10265 CJK02Y 134137472 IC50 = 4170 nM T10265 C8H3ZQ 134138285 IC50 = 3530 nM T10265 CPV75T 134138536 IC50 = 260 nM T10265 C0RD8X 134139097 IC50 = 290 nM T10265 CR4FX3 134139758 IC50 = 1220 nM T10265 C7ZV9I 134140815 IC50 = 1220 nM T10265 CBA5T8 134141183 IC50 = 7550 nM T10265 C06AXV 134142495 IC50 = 0.38 nM T10265 CY8XW3 134142695 IC50 = 2270 nM T10265 C6RO4F 134147146 IC50 > 30000 nM T10265 CIZ95O 134148810 IC50 = 340 nM T10265 CGS1W0 134149697 IC50 = 2690 nM T10265 CJ2T3L 134150878 IC50 = 320 nM T10265 C4SH8R 134153502 IC50 = 1290 nM T10265 C54FXD 134957362 IC50 > 10000 nM T10265 C3R8SE 135457869 IC50 > 10000 nM T10265 C4ASW0 135544141 IC50 = 3800 nM T10265 C1RK8U 135815296 Ki = 8.9 nM T10265 CTX54Z 135896326 IC50 > 10000 nM T10265 C12UMG 136059728 IC50 > 1000 nM T10265 C2VO1H 136132220 Ki = 21.4 nM T10265 C8PG9Q 136132221 Ki = 11 nM T10265 CUI4W9 136132222 Ki = 5.2 nM T10265 CST26Q 136132223 Ki = 11.6 nM T10265 CQ27TM 136132224 Ki = 533 nM T10265 CMIY85 136132225 Ki = 7.6 nM T10265 C7J3IT 136132226 Ki = 42.8 nM T10265 CT3IC8 136132227 Ki = 430 nM T10265 CYM29K 136132228 Ki = 13 nM T10265 CEM5N1 136132229 Ki > 50000 nM T10265 C4V5AD 136132230 Ki = 21.9 nM T10265 CJC0X9 136132231 Ki = 269 nM T10265 COA9T2 136132232 Ki = 10.3 nM T10265 CQ50CG 136132233 Ki = 33 nM T10265 CY50JV 136132234 Ki = 9.8 nM T10265 C28IYL 136132235 Ki = 17.3 nM T10265 CHW75A 136132236 Ki = 9.7 nM T10265 C9GA2W 136132237 Ki = 71.3 nM T10265 C39MDZ 136132238 Ki = 5.8 nM T10265 CW3FM6 136132239 Ki = 11 nM T10265 C5XBZ6 136132240 Ki = 46.9 nM T10265 CU8RC1 136132241 Ki = 26.6 nM T10265 C5NVZ9 136132242 Ki = 18.9 nM T10265 CF31SZ 136132243 Ki = 9.5 nM T10265 C93HEW 136241010 IC50 = 3310 nM T10265 CH30RE 136260531 IC50 = 5.1 nM T10265 C1WD2A 137349131 Ki = 3162.28 nM T10265 CPM38K 137349704 Ki = 630.96 nM T10265 CIM39F 137631787 IC50 = 18400 nM T10265 CBKH04 137632496 IC50 > 100000 nM T10265 CZ5U2B 137633405 IC50 = 45100 nM T10265 CUQX48 137633685 IC50 = 88700 nM T10265 COX0Y5 137633836 IC50 = 28900 nM T10265 C1UTB5 137634455 IC50 = 85600 nM T10265 CEFR52 137635447 IC50 = 6050 nM T10265 C3I6OE 137636108 IC50 = 54800 nM T10265 C9P3UR 137637125 IC50 = 1950 nM T10265 CHYD76 137637146 IC50 = 6700 nM T10265 CS81VD 137637205 IC50 = 240 nM T10265 C92JAF 137637269 IC50 = 1350 nM T10265 C24FLU 137639441 IC50 = 75800 nM T10265 CYJ75P 137640039 IC50 = 2100 nM T10265 CM08AB 137642277 IC50 = 35 nM T10265 C1RPY9 137642586 IC50 = 15800 nM T10265 C7IA8E 137642910 IC50 = 54800 nM T10265 C0AXK5 137642993 IC50 = 22360 nM T10265 C9QG5S 137644770 IC50 = 39700 nM T10265 CH7QG9 137645629 IC50 = 3200 nM T10265 CS0LW7 137646240 IC50 = 8400 nM T10265 CYK2A9 137646728 IC50 = 2620 nM T10265 C2YQR0 137648937 IC50 = 52100 nM T10265 COGR93 137649084 IC50 = 4100 nM T10265 CM8AI0 137649402 IC50 = 9800 nM T10265 C2NXY7 137649733 IC50 = 5800 nM T10265 CQR23F 137650625 IC50 = 40800 nM T10265 C2TZM4 137650925 IC50 = 600 nM T10265 CE69UN 137651372 IC50 = 1300 nM T10265 CLN2U7 137652270 IC50 = 3500 nM T10265 C7X5RC 137654874 IC50 = 5300 nM T10265 CR8E9J 137655231 IC50 = 8180 nM T10265 C0C8NA 137655305 IC50 = 5900 nM T10265 COR2X5 137657511 IC50 = 4100 nM T10265 C3EUK9 137658944 IC50 = 17500 nM T10265 CD8SV1 137660145 IC50 = 58700 nM T10265 CZ74EQ 137660888 IC50 = 4500 nM T10265 CA4J9M 137662320 IC50 = 2060 nM T10265 CRD9Z0 138454907 Ki = 794.33 nM T10265 C8XCM3 138753179 Ki = 316.23 nM T10265 C3BMU6 138753640 Ki = 1000 nM T10265 CO2T5B 138753641 Ki = 794.33 nM T10265 CKRL80 138753642 Ki = 630.96 nM T10265 CVX8G7 138857410 Ki = 398.11 nM T10265 C56CGS 141732269 IC50 > 10000 nM T10265 C6RV9G 141732270 IC50 > 10000 nM T10265 C5NQO6 141732271 IC50 > 10000 nM T10265 CYC4N7 141732272 IC50 = 680 nM T10265 C8I3UK 141732274 IC50 > 10000 nM T10265 C21MEY 141732275 IC50 > 10000 nM T10265 COD59W 141732278 IC50 > 10000 nM T10265 CAP0M8 141732281 IC50 > 100000 nM T10265 C8LBI3 141732282 IC50 = 340 nM T10265 CK9IN8 141732285 IC50 = 2300 nM T10265 C0C4RF 141732286 IC50 > 10000 nM T10265 CNYA07 142592630 IC50 = 61 nM T10265 CX7IJ4 142592631 IC50 = 252 nM T10265 C3TY8Q 142592632 IC50 = 73 nM T10265 C1S7HV 142592633 IC50 = 67 nM T10265 CN3OC2 142592634 IC50 = 15 nM T10265 CP1KB6 142592635 IC50 = 95 nM T10265 CY64NR 142592636 IC50 = 44 nM T10265 C1VDW5 142592637 IC50 = 150 nM T10265 C36OPJ 142592638 IC50 = 367 nM T10265 CSU21G 142592639 IC50 = 477 nM T10265 C5LD3R 142592640 IC50 = 238 nM T10265 CJV32Q 142592643 IC50 = 506 nM T10265 CL0K9J 142592644 IC50 = 881 nM T10265 CZV3M0 142592645 IC50 = 189 nM T10265 C5D7TR 142592646 IC50 = 166 nM T10265 CH4X0J 142592647 IC50 = 239 nM T10265 C7VKY2 142592648 IC50 = 634 nM T10265 C83XNL 142592649 IC50 = 31 nM T10265 CP35HV 142592650 IC50 = 195 nM T10265 C7XZB1 142592652 IC50 = 61 nM T10265 C5W9NS 142592660 IC50 = 178 nM T10265 CH9SB7 142592661 IC50 = 266 nM T10265 C82KMZ 142592663 IC50 = 833 nM T10265 C9SH7Y 145949856 IC50 = 2970 nM T10265 C4PEM2 145950282 IC50 = 50300 nM T10265 C0MT4D 145950945 IC50 = 4100 nM T10265 CZ6FW8 145951897 IC50 = 39900 nM T10265 CL2X1V 145952205 IC50 = 79600 nM T10265 CM68FH 145952334 IC50 = 21100 nM T10265 CD8C1Z 145952416 IC50 = 22200 nM T10265 C0BQ7T 145952944 IC50 = 9400 nM T10265 C0MO2L 145953102 IC50 = 17100 nM T10265 C3JY9H 145953411 IC50 = 2600 nM T10265 C9EC6O 145955031 IC50 = 6100 nM T10265 C3I4YU 145955201 IC50 = 66300 nM T10265 CBS1F9 145955232 IC50 = 2600 nM T10265 CL03PE 145955854 IC50 = 1500 nM T10265 CK6RA0 145957385 IC50 = 70900 nM T10265 C3B5FN 145957516 IC50 = 25700 nM T10265 CD5R3O 145957727 IC50 = 18900 nM T10265 CK1D0W 145957834 IC50 = 46800 nM T10265 CA10IM 145958334 IC50 = 30900 nM T10265 C9JLQ0 145959620 IC50 = 58400 nM T10265 CRX30Z 145959784 IC50 = 9400 nM T10265 CWUZ70 145960159 IC50 = 15200 nM T10265 CJ42NA 145963856 IC50 = 8350 nM T10265 C5CL3K 145964282 IC50 = 1400 nM T10265 C0IC6F 145964309 IC50 > 200000 nM T10265 CCM4E7 145964412 IC50 > 200000 nM T10265 CG12JY 145964431 Ki = 6309.57 nM T10265 CK4YG1 145964495 Ki = 1000 nM T10265 CNGR41 145964560 IC50 = 5.23 nM T10265 CYCS20 145964965 IC50 = 1.26 nM T10265 CM3YN0 145964973 Ki = 50118.72 nM T10265 C2PKI8 145964993 IC50 = 8050 nM T10265 CEV2C0 145965057 IC50 = 4400 nM T10265 CYS17B 145965099 IC50 = 1050 nM T10265 CEGI75 145965101 IC50 = 0.57 nM T10265 CW6R4V 145965268 IC50 = 2850 nM T10265 CDEA40 145965806 Ki = 6309.57 nM T10265 CA6H9G 145965897 IC50 = 19650 nM T10265 CZF69G 145966063 IC50 = 37000 nM T10265 C1H4RT 145966342 IC50 = 51800 nM T10265 CK34EQ 145966780 Ki = 3162.28 nM T10265 C5T8OJ 145966852 Ki = 3981.07 nM T10265 CDYL80 145967203 IC50 = 0.68 nM T10265 CQXK82 145967280 IC50 = 8.67 nM T10265 C18ZXP 145967282 IC50 = 2.28 nM T10265 C1QV4Y 145967438 IC50 = 12720 nM T10265 C4JR7O 145967554 IC50 > 200000 nM T10265 C6YXM2 145968230 IC50 = 26900 nM T10265 C5MV2D 145969186 IC50 = 1.6 nM T10265 C7BVL0 145969367 IC50 = 16350 nM T10265 CH17DI 145969394 Ki = 3162.28 nM T10265 CL4X7Z 145970756 Ki = 630.96 nM T10265 CB75LQ 145970776 Ki = 1995.26 nM T10265 CVIW58 145971796 Ki = 1995.26 nM T10265 CK2Q1M 145972042 IC50 = 7700 nM T10265 CF40VI 145972847 IC50 = 20460 nM T10265 C06GYZ 145972902 IC50 = 66900 nM T10265 CL46GW 145973062 IC50 = 3100 nM T10265 CUD96Q 145973205 Ki = 3981.07 nM T10265 CE1DL4 145973269 IC50 = 1.17 nM T10265 CFS8N5 145973376 IC50 = 3000 nM T10265 CXY3H9 145973870 IC50 = 16200 nM T10265 CZAJ58 145973921 IC50 = 1620 nM T10265 CY2R1M 145974127 IC50 = 12500 nM T10265 CC7HN2 145974174 IC50 = 880 nM T10265 CZEW75 145974259 IC50 = 5500 nM T10265 CJQH60 145974519 Ki = 2511.89 nM T10265 CL0ZP8 145974645 IC50 = 7400 nM T10265 CF9O2T 145974687 Ki = 10000 nM T10265 C0JQ3V 145974692 IC50 > 200000 nM T10265 CLV25P 145974711 IC50 = 44000 nM T10265 C9RGV1 145974955 IC50 = 3250 nM T10265 CNBC60 145975232 IC50 > 200000 nM T10265 C06YIC 145975272 Ki = 31.62 nM T10265 C2GIR6 145975414 IC50 = 11020 nM T10265 CI6AV5 145975668 IC50 = 1.87 nM T10265 CDKI37 145975800 IC50 = 1.06 nM T10265 C6W7RB 145975941 IC50 = 31100 nM T10265 C7QHD6 145976252 IC50 > 50000 nM T10265 CS1V9B 145976314 IC50 = 47800 nM T10265 CP9R8Z 145976467 IC50 = 2380 nM T10265 C5NR0W 145976583 IC50 = 18350 nM T10265 C0WIK2 145976775 Ki = 12589.25 nM T10265 CYR25Q 145976879 Ki = 7943.28 nM T10265 CHP1E6 145976908 IC50 = 1.22 nM T10265 CN61GR 145977095 IC50 = 70800 nM T10265 C8MT9S 145977100 IC50 = 3420 nM T10265 CN47BX 145977141 Ki = 2511.89 nM T10265 CI58DJ 145977392 Ki = 2511.89 nM T10265 CD09US 145977528 IC50 = 116100 nM T10265 CTZ6O9 145977634 IC50 = 1900 nM T10265 CZ50HJ 145977998 IC50 = 7900 nM T10265 CH2N8C 145978004 IC50 > 50000 nM T10265 CVNQ81 145978210 Ki = 158.49 nM T10265 CK1BR0 145978345 IC50 = 950 nM T10265 CN9K3J 145978566 IC50 = 1.28 nM T10265 CAM63C 145978719 IC50 = 2.92 nM T10265 CG0C4K 145978810 IC50 = 0.75 nM T10265 CKOT32 145978829 IC50 = 1800 nM T10265 CO3DQ9 145978852 IC50 > 50000 nM T10265 CZC61L 145978996 IC50 > 200000 nM T10265 CM8A5X 145979217 IC50 = 20200 nM T10265 C0JRK5 145980304 IC50 > 200000 nM T10265 C3GL0U 145980967 IC50 = 45300 nM T10265 CV7G5F 145981927 IC50 = 87490 nM T10265 C7BP2S 145981946 IC50 > 200000 nM T10265 CK45RB 145981967 IC50 = 8400 nM T10265 C42VHC 145982018 IC50 = 16830 nM T10265 C5RCY6 145982932 IC50 > 200000 nM T10265 C4HJ5U 145983187 IC50 = 7200 nM T10265 C7B0CK 145983920 IC50 = 52400 nM T10265 CT1L8E 145986656 IC50 = 42460 nM T10265 C1TU2D 145986784 IC50 = 5430 nM T10265 CU0H4T 145986885 IC50 = 20900 nM T10265 CAS90U 145986925 IC50 = 17840 nM T10265 C3SV8R 145987119 IC50 > 200000 nM T10265 C6K2MS 145987191 IC50 = 1700 nM T10265 C9TYX0 145987253 IC50 = 15400 nM T10265 CM6P3Z 145987468 IC50 = 32290 nM T10265 C7C3KG 145987995 IC50 = 222 nM T10265 C0ODP3 145988021 IC50 > 200000 nM T10265 C25WHX 145988690 IC50 = 14690 nM T10265 C35GWH 145989417 IC50 = 109820 nM T10265 CY75SD 145989570 IC50 > 200000 nM T10265 CRP0I2 145989866 IC50 = 70300 nM T10265 CUK86E 145989957 IC50 = 21140 nM T10265 CV9BP4 145990259 IC50 > 200000 nM T10265 CAPB90 145990360 IC50 = 51100 nM T10265 CB6MV7 145990536 IC50 = 14500 nM T10265 C6NHE1 145990687 IC50 > 200000 nM T10265 C7X8AF 145990697 IC50 = 35900 nM T10265 CIR0A5 145991365 IC50 = 62700 nM T10265 COSL82 145992781 IC50 > 200000 nM T10265 C8CSM5 145992787 IC50 > 200000 nM T10265 CPD5L1 145993291 IC50 = 3900 nM T10265 C59VKM 145993568 IC50 = 74 nM T10265 CG5E3A 145993704 IC50 > 200000 nM T10265 C42OZA 145993939 IC50 = 3200 nM T10265 CI7H3T 145994146 IC50 > 200000 nM T10265 CHJ79V 145997874 IC50 = 8 nM T10265 C3O6AQ 155511651 Ki = 630.96 nM T10265 C04SNH 155512285 IC50 > 100000 nM T10265 CS8DT7 155513046 IC50 = 4100 nM T10265 CTP50A 155513604 Ki = 199.53 nM T10265 CQ6F8J 155514145 Ki = 630.96 nM T10265 C1JSC7 155514219 Ki = 794.33 nM T10265 CT9W1I 155516764 IC50 = 4670 nM T10265 C4N8ZM 155517074 Ki = 398.11 nM T10265 C18BIY 155518011 Ki = 251.19 nM T10265 CIV9H6 155518343 Ki = 501.19 nM T10265 C03WPT 155518716 IC50 = 1040 nM T10265 C7JPT1 155519178 IC50 = 3960 nM T10265 CL8CU6 155521936 IC50 = 1650 nM T10265 CDK3B5 155522558 Ki = 398.11 nM T10265 CMZG78 155523502 Ki = 630.96 nM T10265 C4YQZ5 155525638 IC50 = 440 nM T10265 CD0T4G 155527425 IC50 = 3700 nM T10265 C4OQI1 155528367 IC50 = 16460 nM T10265 C8O6RT 155529515 Ki = 316.23 nM T10265 CT85RG 155530589 IC50 = 220 nM T10265 CJCD73 155531859 IC50 > 10000 nM T10265 CZ91HU 155533144 IC50 = 390 nM T10265 C4GQO3 155534561 IC50 = 3860 nM T10265 C5Z7PM 155535141 Ki = 501.19 nM T10265 CG07OY 155535903 Ki = 794.33 nM T10265 CQ30UY 155535906 IC50 = 29360 nM T10265 CR9V1W 155536560 Ki = 794.33 nM T10265 CT8MU5 155537132 IC50 > 10000 nM T10265 CK4B8R 155537321 IC50 = 5970 nM T10265 C8SZP7 155540165 Ki = 398.11 nM T10265 C0KTQ9 155542215 Ki = 1584.89 nM T10265 C84JYS 155542300 Ki = 1258.93 nM T10265 C8N4KT 155542744 Ki = 501.19 nM T10265 C4JKX7 155542965 IC50 = 5580 nM T10265 CLWO73 155543362 IC50 > 100000 nM T10265 C5WK6B 155543774 Ki = 501.19 nM T10265 CAK8N3 155543874 IC50 = 18360 nM T10265 CEMT29 155545548 IC50 = 36480 nM T10265 CL92GR 155546391 IC50 = 9740 nM T10265 CNPQ31 155548321 IC50 = 20460 nM T10265 CD6K2Y 155548709 IC50 = 4250 nM T10265 CKJ1S2 155550312 Ki = 316.23 nM T10265 C8V4AW 155551577 IC50 = 8320 nM T10265 C5DP1T 155552281 IC50 = 940 nM T10265 C24DCR 155552652 IC50 = 3500 nM T10265 CN1R8L 155552930 IC50 = 3880 nM T10265 CK5VS2 155556362 IC50 > 10000 nM T10265 C8L0OY 155559141 Ki = 794.33 nM T10265 C0JOE4 155560799 Ki = 1000 nM T10265 CTL6O7 155562866 IC50 = 1850 nM T10265 C3CR6S 155563411 IC50 = 43160 nM T10265 C9JHD6 155563445 IC50 = 790 nM T10265 C7KBJ3 155563967 IC50 = 7530 nM T10265 CY4S1X 155564743 IC50 = 1850 nM T10265 CW9KA7 155565974 Ki = 1258.93 nM T10265 C0CH3Y 155566295 IC50 = 210 nM T10265 CI8WV3 155567794 IC50 = 2030 nM T10265 CB5JS1 155568212 IC50 = 1980 nM T10265 D00MBG 2921148 IC50 = 1800 nM T10265 D00ZGW 46883841 IC50 = 3981.07 nM T10265 D01NVD 46830196 IC50 > 2511.89 nM T10265 D01RUN 448055 IC50 = 39.81 nM T10265 D09RKU 46239428 Ki > 10000 nM T10265 D0D6MC 1150897 IC50 > 200000 nM T10265 D0JD4C 9853498 IC50 = 0.5 nM T10265 D0K4HG 9819356 IC50 = 0.07 nM T10265 D0P2TS 9818682 IC50 = 1500 nM T10265 D0R6MT 3758 IC50 = 28200 nM T10265 D0V1CL 37015 IC50 = 199.53 nM T10265 D0V4WB 149790 IC50 > 16000 nM T10265 D0W7WV 11039077 IC50 = 0.4 nM T10265 D0WU1S 52912189 IC50 = 3981.07 nM T89083 CKA2Q3 8030846 EC50 = 560 nM T89083 CV71BY 11491636 IC50 = 230 nM T89083 C09ZEH 11600631 IC50 = 5000 nM T89083 COW07X 11643706 IC50 = 900 nM T89083 CLW30D 13633114 EC50 = 6430 nM T89083 C7JVW2 25157439 IC50 = 460 nM T89083 C1DSU6 44405462 IC50 = 950 nM T89083 C8VJ5F 44405524 IC50 = 1250 nM T89083 CF5WB8 44405603 IC50 = 2150 nM T89083 CBH7W9 44405604 IC50 = 5200 nM T89083 CA0GC9 44405661 IC50 = 22000 nM T89083 C12EAM 44405768 IC50 = 6460 nM T89083 C0Q5XC 44405780 IC50 = 6900 nM T89083 CBZ97N 44405822 IC50 = 1600 nM T89083 CN23KH 44589027 IC50 = 240 nM T89083 CBNO65 44589028 IC50 = 900 nM T89083 CHG12U 46201898 IC50 = 1200 nM T89083 C7X3PH 46205782 IC50 = 48 nM T89083 CDG83H 46732368 EC50 = 350 nM T89083 C9SFC7 46732463 EC50 = 8550 nM T89083 CBE2P6 54679465 EC50 = 300 nM T89083 C3W4DU 56655503 EC50 = 0.26 nM T89083 CB3AF0 56849710 EC50 = 0.45 nM T89083 CWC72K 56849711 EC50 = 1 nM T89083 CU7Q1J 56849712 EC50 = 0.87 nM T89083 C9TX4L 56849854 EC50 > 1000 nM T89083 C37INL 56849985 EC50 = 6.48 nM T89083 CSAM54 56849987 EC50 = 0.56 nM T89083 CG3IS5 56850128 EC50 = 1.47 nM T89083 C8X4NH 56850131 EC50 > 1000 nM T89083 CT1J9P 56850266 EC50 = 2.11 nM T89083 C3GCL2 56850401 EC50 = 1.55 nM T89083 CV0HU7 56850403 EC50 = 3.23 nM T89083 CX95CN 56850406 EC50 = 1.95 nM T89083 C3UHQ9 56850535 EC50 = 1.86 nM T89083 CW4ZC5 56850682 EC50 = 3.63 nM T89083 CSHE59 56850818 EC50 > 1000 nM T89083 C25HAU 56850822 EC50 > 1000 nM T89083 CUAK61 56850940 EC50 > 1000 nM T89083 CQJ4W0 56851062 EC50 > 1000 nM T89083 C4K8NM 56851182 EC50 > 1000 nM T89083 CLT65O 56851306 EC50 > 1000 nM T89083 CQH8R9 56851450 EC50 > 1000 nM T89083 C35ONK 57384785 EC50 = 1.01 nM T89083 C4ZY6M 57384786 EC50 = 1.64 nM T89083 CQ5Z0D 57384787 EC50 = 3.8 nM T89083 C1Z9CB 57384789 EC50 = 4.5 nM T89083 CU30HE 57388031 EC50 = 5.52 nM T89083 CB1VQ8 57388036 EC50 = 4.79 nM T89083 C4Y5XA 57740266 EC50 = 23 nM T89083 CH29GF 71258526 IC50 > 10000 nM T89083 CIB14T 71451937 Ki = 25 nM T89083 CPCT40 71451938 EC50 = 78 nM T89083 C83LQK 71453783 EC50 = 25 nM T89083 CZDG94 71457280 EC50 = 3.7 nM T89083 C2KRU3 71457309 EC50 = 56 nM T89083 CKQ03G 71462640 EC50 = 20 nM T89083 CGJ0Q1 118719088 Ki = 11 nM T89083 C45BQH 132585194 EC50 > 100000 nM T89083 CAVF95 137553173 EC50 = 0.11 nM T89083 CTP9M8 145968052 IC50 = 4651 nM T89083 COQ29Y 145968118 IC50 = 4363 nM T89083 C4T7FK 145968297 IC50 = 1682 nM T89083 CJ01EH 145968400 IC50 = 4755 nM T89083 CR8SB5 145968508 IC50 = 3373 nM T89083 CY6GD5 145969059 IC50 = 7519 nM T89083 CYQZ05 145969942 IC50 = 3938 nM T89083 CP50WV 145970164 IC50 = 1962 nM T89083 CE41IX 145987954 IC50 = 6427 nM T89083 CAKE87 149687120 EC50 = 1000 nM T89083 CRJ74Z 150370253 EC50 = 1350 nM T89083 CT2CO6 150457654 EC50 = 3000 nM T89083 C0GR6S 151417654 EC50 = 5000 nM T89083 CAC0J5 151485696 EC50 = 1450 nM T89083 CL7F2W 151543599 EC50 = 320 nM T89083 CAM64K 152550631 EC50 = 3090 nM T89083 CO94FB 152580191 EC50 = 45240 nM T89083 C1QR9N 152598982 EC50 = 6630 nM T89083 C67ORV 155514087 EC50 = 46.16 nM T89083 CN6IC3 155515837 EC50 = 0.304 nM T89083 C9L5GP 155519718 EC50 = 160 nM T89083 C3SNM6 155524646 EC50 = 150.6 nM T89083 CISL79 155528194 EC50 = 0.609 nM T89083 CAI06Z 155528951 EC50 = 3460 nM T89083 CUM0D7 155530294 EC50 = 161.01 nM T89083 CO8T1L 155533032 EC50 = 4590 nM T89083 C3YD6A 155534493 EC50 = 450 nM T89083 C7KV8W 155535367 EC50 = 11820 nM T89083 CL6A9D 155536490 EC50 = 16380 nM T89083 C74LZY 155537225 EC50 = 14160 nM T89083 C2NRE1 155548273 EC50 = 1.162 nM T89083 CW2V9Z 155548681 EC50 = 1330 nM T89083 CHSC79 155553471 EC50 = 0.383 nM T89083 C1Y6NK 155555507 EC50 = 0.281 nM T89083 CE1Q2L 155558171 EC50 = 0.468 nM T89083 CU7S9Z 155559013 EC50 = 155.69 nM T89083 CQ4I7V 155562153 EC50 = 4.445 nM T89083 C6H2TX 155562332 EC50 = 17.38 nM T89083 CSW73J 155564215 EC50 = 22.96 nM T89083 D02TVS 985 IC50 = 5000 nM T89083 D08OBF 11005 IC50 = 5000 nM T72335 D05JNI 8378 Ki = 500 nM T72335 D0L5WM 2157 IC50 = 3500 nM T72335 D0R9BG 1990 IC50 = 11400000 nM T72335 D0Y4JJ 2351 IC50 = 4800 nM T72335 C49BCY 1570 IC50 = 5000000 nM T72335 CQ86IR 47363 IC50 = 49000 nM T72335 C47RSL 52603 IC50 = 43000 nM T72335 CEU84H 67070 Ki = 560 nM T72335 C7P3UR 69975 IC50 = 5000000 nM T72335 C8BT0E 206023 IC50 > 100000 nM T72335 C50TDK 234080 IC50 > 100000 nM T72335 CCKZ79 668744 Ki = 1500 nM T72335 CM7S8X 670897 IC50 = 60000 nM T72335 CEUN62 689246 IC50 = 4365.16 nM T72335 C0ER8S 767161 Ki = 900 nM T72335 CDVJ42 767163 Ki = 1600 nM T72335 CRAE16 769062 IC50 > 100000 nM T72335 CE10WO 776842 Ki = 5600 nM T72335 CQ2R0M 1011274 Ki = 900 nM T72335 CZDL61 1041898 IC50 = 2089.3 nM T72335 C9YKQ5 1201190 IC50 = 79400 nM T72335 C7P1UO 1201257 Ki = 3300 nM T72335 CJH7F4 1204542 IC50 = 16595.87 nM T72335 CNOQ24 1204544 IC50 = 891.25 nM T72335 C1PB2M 1269164 IC50 = 30700 nM T72335 C1CWQ3 1269183 IC50 = 29900 nM T72335 C2PRY6 1269450 Ki = 2700 nM T72335 CI0YJ3 1270226 IC50 = 50000 nM T72335 CN35KL 1273153 IC50 = 21300 nM T72335 CCO87V 1286537 IC50 = 1698.24 nM T72335 CT35RG 1713267 IC50 = 260 nM T72335 CD2GP3 1730599 IC50 = 300 nM T72335 C3M7AE 2009854 IC50 = 3100 nM T72335 CK8Z9W 2140081 IC50 = 850 nM T72335 CO4AB7 2264784 Ki = 5400 nM T72335 C0LF2Z 2275298 IC50 > 100000 nM T72335 C0HP6Q 2735376 IC50 > 100000 nM T72335 C43VPR 2735416 IC50 > 100000 nM T72335 CSG17P 2809632 Ki = 7800 nM T72335 C28QWD 2880808 IC50 > 100000 nM T72335 C6QFC2 2921978 IC50 = 15900 nM T72335 C1D2XG 4330580 Ki = 1800 nM T72335 CC5O4E 4369384 Ki = 24 nM T72335 CQWL43 5039074 Ki = 2900 nM T72335 CZ6A5E 5286524 IC50 > 100000 nM T72335 CY36BO 5289928 IC50 > 100000 nM T72335 CT8I1B 5292405 Ki = 3100 nM T72335 CFVH71 5334847 IC50 > 100000 nM T72335 C4H0RI 5339251 IC50 = 20900 nM T72335 C9SE5W 5348600 Ki = 570 nM T72335 CLD0C6 5348879 Ki = 7200 nM T72335 CF1P5H 5430316 Ki = 900 nM T72335 C6L9AJ 5499083 IC50 = 31700 nM T72335 C8NX4U 5499839 Ki = 1600 nM T72335 CAB14K 5713760 Ki = 6600 nM T72335 CNCU03 5733576 IC50 = 29600 nM T72335 C8OYI5 5738327 IC50 > 100000 nM T72335 CU51FT 5738908 IC50 > 100000 nM T72335 C8U1EX 5754107 IC50 > 100000 nM T72335 C4UK9R 5765823 IC50 > 100000 nM T72335 C10BFH 5827835 IC50 = 190 nM T72335 CZ1XU5 5876194 Ki = 800 nM T72335 CI05ML 5915017 IC50 > 100000 nM T72335 C7EVJ1 5931873 IC50 > 100000 nM T72335 CDI23X 5941957 IC50 = 74000 nM T72335 CFH67Y 5971874 IC50 = 5600 nM T72335 C4J3PG 6250177 Ki = 4200 nM T72335 CA0G1L 6539635 IC50 = 740 nM T72335 CBHG28 6539636 IC50 = 3235.94 nM T72335 CB1HZ8 6539637 IC50 = 1584.89 nM T72335 CW4CD3 6539638 IC50 = 72400 nM T72335 C5S3CN 6539639 IC50 = 10000 nM T72335 CDX13Q 6539640 IC50 = 5000 nM T72335 CV46UF 6539641 IC50 = 4365.16 nM T72335 CGEC06 6539642 IC50 = 5888.44 nM T72335 CTWE21 6539646 IC50 = 1288.25 nM T72335 CAMX42 6539647 IC50 = 1200 nM T72335 CYE4A1 6539648 IC50 = 2290.87 nM T72335 CI9JL0 6539649 IC50 = 22387.21 nM T72335 CW6PI9 6539650 IC50 = 5600 nM T72335 CI86PQ 6539651 IC50 = 900 nM T72335 CN7I0E 6539652 IC50 > 20000 nM T72335 CZF83S 6539653 IC50 > 40000 nM T72335 CN0Q7S 6539654 IC50 > 40000 nM T72335 C0G9KA 6539655 IC50 = 3100 nM T72335 CV3SC8 6539656 IC50 = 2100 nM T72335 C9RI1H 6539657 IC50 = 19100 nM T72335 CXPL32 6539658 IC50 = 1100 nM T72335 CUS27J 6539659 IC50 = 6600 nM T72335 C2E9AO 6539660 IC50 = 2800 nM T72335 CMG4W6 6539661 IC50 = 290 nM T72335 CEOY78 6539662 IC50 = 3000 nM T72335 CVNO37 6539663 IC50 = 400 nM T72335 CE36WO 6539664 IC50 = 120 nM T72335 CJH7B8 6539665 IC50 > 20000 nM T72335 CIN31Z 6539666 IC50 = 5180 nM T72335 CAE34V 6539667 IC50 = 11880 nM T72335 C1R3VP 6539668 IC50 = 16600 nM T72335 CMB59U 6539669 IC50 > 20000 nM T72335 CQEF36 6539670 IC50 > 40000 nM T72335 CZM4F6 6539671 IC50 > 40000 nM T72335 C63KTU 6539672 IC50 > 20000 nM T72335 C5XKI4 6539673 IC50 = 2760 nM T72335 CMA32G 6539674 IC50 = 1640 nM T72335 C8NUS2 6539675 IC50 = 3740 nM T72335 C0FCO5 6539676 IC50 = 1310 nM T72335 C85ODN 6539677 IC50 = 1310 nM T72335 CE4TP3 6539678 IC50 = 810 nM T72335 C2M5AQ 6539679 IC50 = 500 nM T72335 COL78Q 6539680 IC50 = 100 nM T72335 C1M9PW 6539681 IC50 = 70 nM T72335 C7U5FE 6539682 IC50 = 300 nM T72335 C3I2AS 6539683 IC50 = 730 nM T72335 CQB2S6 6539684 IC50 = 670 nM T72335 C0JL1I 6539685 IC50 = 64 nM T72335 C6G4NS 6539686 IC50 = 42 nM T72335 C3HKC7 6539687 IC50 = 50 nM T72335 CK94EY 6539689 IC50 = 67 nM T72335 CB1P9G 6539690 IC50 = 67 nM T72335 CLQ32E 6539691 IC50 = 51 nM T72335 CIG2S5 6539692 IC50 = 65 nM T72335 C1X8QT 6602516 IC50 = 37 nM T72335 CJ79SO 6602517 IC50 = 7470 nM T72335 C2Q7US 6602518 IC50 = 57 nM T72335 C3OT2H 6602520 IC50 = 40 nM T72335 CG2A7X 7028541 Ki = 1100 nM T72335 CY98UW 9638046 IC50 = 26600 nM T72335 CZ32TB 9678168 IC50 = 25600 nM T72335 CXWO50 9688146 IC50 = 29700 nM T72335 CC4WG3 9957228 Ki = 700 nM T72335 C1M7UG 10383623 IC50 = 75 nM T72335 CJ5SU9 11328354 Ki = 500 nM T72335 CA5P8H 11355488 IC50 = 204000 nM T72335 C8N2MW 11579107 IC50 = 2900 nM T72335 CUIM84 11628682 Ki = 65 nM T72335 CP1V8F 12207688 IC50 = 35000 nM T72335 CM48AT 15133398 IC50 > 100000 nM T72335 CUQG04 16130642 Ki = 365 nM T72335 C5YG0U 16198696 Ki = 381 nM T72335 CW8IJ4 17432052 IC50 > 100000 nM T72335 CB68QY 20831578 IC50 = 16500 nM T72335 CW7ET4 23645946 Ki = 5000 nM T72335 CW6FO4 23645947 Ki = 5200 nM T72335 C78DHE 23645948 Ki = 10900 nM T72335 CMZ5S7 23645949 Ki = 24300 nM T72335 C7KE6P 23645950 Ki = 5600 nM T72335 CJY68O 23645951 Ki = 5300 nM T72335 C8V3AX 23645952 Ki = 10200 nM T72335 C4R2DA 23645953 Ki = 700 nM T72335 C7TGE0 23645954 Ki = 8800 nM T72335 C0A1PD 23645955 Ki = 7700 nM T72335 C9JP3X 23645956 Ki = 8700 nM T72335 CT3CV0 23645957 Ki = 3100 nM T72335 CM2A0D 23645958 Ki = 9200 nM T72335 CWN3I4 23645959 Ki = 1500 nM T72335 C4UEM5 24871537 Ki = 0.24 nM T72335 CP2L5B 24871655 Ki = 0.13 nM T72335 CUI81J 24873445 Ki = 3 nM T72335 CE73LG 24949066 Ki = 380 nM T72335 C1GVE0 24990995 Ki = 2.4 nM T72335 CNXA45 24991001 Ki = 0.39 nM T72335 C8B0JT 24991002 Ki = 0.71 nM T72335 CUT8N4 24991363 Ki = 9.5 nM T72335 CW2BC7 25007684 Ki = 0.05 nM T72335 C2MK1H 25007685 Ki = 30.4 nM T72335 CX1MC0 25007686 Ki = 273 nM T72335 CZ94HL 25007687 Ki = 0.62 nM T72335 CGOY89 25134297 Ki = 11 nM T72335 CLD79X 25164605 Ki = 1.1 nM T72335 CM21PS 40669841 IC50 > 100000 nM T72335 C8TW6U 44219671 IC50 = 6600 nM T72335 CI9V6D 44219672 Ki = 1000 nM T72335 CLF59H 44406615 IC50 > 100000 nM T72335 CYH19P 44406683 IC50 = 500 nM T72335 CRDX58 44407604 IC50 = 48 nM T72335 C56DYC 44407799 IC50 = 450 nM T72335 CU3O2E 44407810 IC50 = 17000 nM T72335 CH6KR2 44409116 Ki = 4100 nM T72335 CNF6R7 44409117 Ki = 31400 nM T72335 C1G6YT 44409119 Ki = 10700 nM T72335 C1H5OC 44409120 Ki = 153700 nM T72335 CUXP25 44409150 Ki = 6600 nM T72335 CA89XB 44409189 Ki = 24800 nM T72335 CFN16L 44409194 Ki = 500 nM T72335 CYG18P 44409381 Ki = 14900 nM T72335 CWC17I 44409382 Ki = 30600 nM T72335 CI3CE1 44409385 Ki = 600 nM T72335 CIP7E1 44415075 Ki = 2400 nM T72335 CMNS58 44415106 IC50 = 14800 nM T72335 CJVG58 44415121 IC50 = 17700 nM T72335 C0THI1 44415189 Ki = 2100 nM T72335 CGDY32 44415219 Ki = 2500 nM T72335 CN07HB 44441631 IC50 = 70000 nM T72335 C8YOL7 45139447 IC50 > 100000 nM T72335 CS12ZJ 45139450 IC50 = 55000 nM T72335 CM85AS 45139630 IC50 > 100000 nM T72335 C72DJF 45139631 IC50 > 100000 nM T72335 C46XBV 45139632 IC50 = 18000 nM T72335 CMVP78 45139633 IC50 > 100000 nM T72335 CXR29W 45139819 IC50 > 100000 nM T72335 CFYJ76 45141625 IC50 > 100000 nM T72335 CQ26MI 45141818 IC50 > 100000 nM T72335 C54IQU 45141819 IC50 = 28000 nM T72335 CAFD63 45141820 IC50 > 100000 nM T72335 CH21VS 45141821 IC50 > 100000 nM T72335 CR7A1J 45142028 IC50 > 100000 nM T72335 COV87J 45142030 IC50 = 51000 nM T72335 C2UTI5 45267101 IC50 = 18000 nM T72335 C4R6JO 45267107 IC50 = 14000 nM T72335 CPZX59 45267121 IC50 = 11000 nM T72335 C4FMY3 45267122 IC50 > 50000 nM T72335 CQB8P7 45267141 IC50 = 16000 nM T72335 C7B3RS 45267157 IC50 = 19000 nM T72335 CJC12N 45267187 IC50 = 9000 nM T72335 CHOV86 45267962 IC50 = 11000 nM T72335 CIPY79 45267963 IC50 > 50000 nM T72335 CTS8B7 45267970 IC50 = 15000 nM T72335 C0FN5C 45267971 IC50 = 10000 nM T72335 C9Z6XR 45267972 IC50 = 27000 nM T72335 C21HBY 45267978 IC50 > 100000 nM T72335 C90FTO 45267979 IC50 > 100000 nM T72335 C2DQ3I 45267980 IC50 = 14000 nM T72335 CW01DI 45267992 IC50 = 19000 nM T72335 CQH29D 45267993 IC50 > 50000 nM T72335 COJ8P7 45268000 IC50 = 16000 nM T72335 CMQ8V9 45268001 IC50 = 100000 nM T72335 CR67PB 45268002 IC50 > 50000 nM T72335 CKY24U 45268004 IC50 = 13000 nM T72335 CA0O7N 45268010 IC50 = 12000 nM T72335 CET0Y8 45268035 IC50 = 3900 nM T72335 CL91FB 45268040 IC50 = 7200 nM T72335 CU57SN 45268840 IC50 = 13000 nM T72335 C40HYE 45268846 IC50 = 19000 nM T72335 CW3FL7 45268847 IC50 = 12000 nM T72335 CO3U8F 45268861 IC50 = 48000 nM T72335 CL23TX 45268862 IC50 = 11000 nM T72335 C8U7AB 45268868 IC50 = 12000 nM T72335 CJ1DG5 45268899 IC50 = 4500 nM T72335 CB63VR 45268903 IC50 = 10000 nM T72335 C30CUT 45268923 IC50 = 8000 nM T72335 CK23TC 45269681 IC50 > 100000 nM T72335 CDZ6U2 45269682 IC50 = 12000 nM T72335 CWAD09 45269689 IC50 > 100000 nM T72335 C5O7PN 45269690 IC50 = 11000 nM T72335 C4BPI2 45269695 IC50 = 8900 nM T72335 C3JN0H 45269696 IC50 > 100000 nM T72335 C0RV7M 45269697 IC50 = 27000 nM T72335 C37KWG 45269701 IC50 = 100000 nM T72335 CQY0R3 45269702 IC50 = 23000 nM T72335 C3QBL7 45269708 IC50 > 100000 nM T72335 CHLJ13 45269709 IC50 = 19000 nM T72335 CRD50S 45269712 IC50 = 12000 nM T72335 C1GDK7 45269713 IC50 = 21000 nM T72335 C4E9CK 45269714 IC50 > 50000 nM T72335 CKQE73 45269719 IC50 = 16000 nM T72335 COS50E 45269720 IC50 = 22000 nM T72335 CVK1A3 45269721 IC50 = 9600 nM T72335 CK50HN 45269722 IC50 > 50000 nM T72335 CB81GA 45269727 IC50 = 24000 nM T72335 CUZ46J 45269728 IC50 > 100000 nM T72335 CMU5N0 45269729 IC50 > 100000 nM T72335 C26XZQ 45269760 Ki = 1700 nM T72335 CBYU69 45269770 IC50 = 3000 nM T72335 C0G5WL 45270516 IC50 = 46000 nM T72335 CXUT59 45270532 IC50 = 19000 nM T72335 C90QNC 45270540 IC50 > 100000 nM T72335 CRO6F4 45270553 IC50 > 50000 nM T72335 CPY83E 45270554 IC50 = 18000 nM T72335 C4JKB8 45270555 IC50 > 100000 nM T72335 CG4KD3 45270564 IC50 = 11000 nM T72335 C4IS9C 45270578 IC50 > 50000 nM T72335 CZ94YD 45270582 IC50 = 11000 nM T72335 C2G8QW 45270596 IC50 = 13000 nM T72335 CS3H8O 45271340 IC50 > 100000 nM T72335 C5RT9W 45271341 IC50 = 8000 nM T72335 CJP34Y 45271346 IC50 = 17000 nM T72335 C9AR8K 45271352 IC50 = 30000 nM T72335 CEUM39 45271357 IC50 = 100000 nM T72335 C59MAP 45271364 IC50 = 17000 nM T72335 CR20UP 45271365 IC50 > 50000 nM T72335 CGIW83 45271378 IC50 = 39000 nM T72335 CQ38RD 45271384 IC50 = 11000 nM T72335 C6Q8ZL 45271400 IC50 = 13000 nM T72335 CR71YC 45271401 IC50 = 13000 nM T72335 CXC4U3 45271405 IC50 = 15000 nM T72335 C5DTC0 45271420 IC50 = 9000 nM T72335 CJO0F6 45271421 IC50 > 50000 nM T72335 C34CMD 45271422 IC50 = 43000 nM T72335 C75AGK 45272234 IC50 = 9400 nM T72335 C5J7QT 45272235 IC50 = 25000 nM T72335 CNC90Y 45272242 IC50 > 100000 nM T72335 C4QFW7 45272244 IC50 = 35000 nM T72335 CKY65P 45272245 IC50 = 22000 nM T72335 CHG43J 45272248 IC50 = 34000 nM T72335 C9BQ7S 45272249 IC50 = 10000 nM T72335 CRV92F 45272254 IC50 = 28000 nM T72335 C3KV2A 45272261 IC50 > 100000 nM T72335 CSJF68 45272275 IC50 = 39000 nM T72335 CB8VX0 45272292 IC50 = 28000 nM T72335 CR37UG 45272303 IC50 = 14000 nM T72335 CZ49LB 45273101 IC50 = 17000 nM T72335 CG9O1M 45273110 IC50 = 11000 nM T72335 CVA13D 45273111 IC50 = 18000 nM T72335 C53JSC 45273112 IC50 > 50000 nM T72335 CS0G3Q 45273114 IC50 > 50000 nM T72335 C8J9QC 45273119 IC50 = 17000 nM T72335 C8D0CP 45273120 IC50 > 100000 nM T72335 CUYM65 45273121 IC50 > 50000 nM T72335 CV0X4O 45273133 IC50 = 9300 nM T72335 CFWH25 45273143 IC50 = 18000 nM T72335 CV43JT 45273155 IC50 = 9000 nM T72335 C17OIV 45273162 IC50 = 30000 nM T72335 CEA8R4 45273163 IC50 = 10000 nM T72335 CF6CV1 45273170 IC50 = 8000 nM T72335 CX2P4E 45273171 IC50 = 8000 nM T72335 CC7XI4 45273178 IC50 = 18000 nM T72335 CDJ5B9 46228743 IC50 > 100000 nM T72335 CF8OK2 46228744 IC50 > 100000 nM T72335 CP36UA 46228780 IC50 = 48000 nM T72335 CJQ78T 46228781 IC50 = 40000 nM T72335 CH2O6D 46228782 IC50 > 100000 nM T72335 CH3O4A 46228783 IC50 > 100000 nM T72335 CGP49Y 46228784 IC50 = 61000 nM T72335 C3ZL8M 46228836 IC50 > 100000 nM T72335 CAR0S9 46228837 IC50 > 100000 nM T72335 CJZA45 46232267 IC50 > 100000 nM T72335 C3PLE6 46232269 IC50 > 100000 nM T72335 C3U8HV 46232270 IC50 > 100000 nM T72335 CYA73D 46232312 IC50 > 100000 nM T72335 C7AU4S 50943150 IC50 > 100000 nM T72335 C2V9DP 50943152 IC50 > 100000 nM T72335 C5D9SV 51397591 IC50 = 7000 nM T72335 CSH41O 52940940 Ki = 122 nM T72335 C6ML8V 52941404 IC50 = 300 nM T72335 C1FAR4 52941405 IC50 = 500 nM T72335 C8O6BH 52941619 Ki = 9.3 nM T72335 CB1AS8 52941676 Ki = 0.44 nM T72335 C8I9RS 52942110 Ki = 7.3 nM T72335 CIO84Q 52942118 Ki = 3.1 nM T72335 C0OG9N 52942165 Ki = 0.3 nM T72335 C9MOW8 52943189 Ki = 8.2 nM T72335 CV52FH 52944453 Ki = 350 nM T72335 C2Q0FR 52944538 Ki = 33 nM T72335 CU7Y1R 52944559 Ki = 1.4 nM T72335 CVX14Y 52945702 Ki = 99 nM T72335 C7ZF6N 52945720 Ki = 118 nM T72335 C20VAX 52945792 Ki = 96 nM T72335 CKF9X8 52945883 Ki = 0.85 nM T72335 CU07MG 52945891 Ki = 0.47 nM T72335 CA48FQ 52945924 Ki = 0.69 nM T72335 C5F0OE 52945932 Ki = 0.41 nM T72335 C3NV4E 52946540 Ki = 115 nM T72335 C7EZ8P 52946921 Ki = 151 nM T72335 C8LC9G 52946940 Ki = 135 nM T72335 C9H5CX 52947005 Ki = 230 nM T72335 C4L9JZ 52947485 IC50 = 700 nM T72335 CM2QU6 52948143 Ki = 42 nM T72335 CED63M 52948249 Ki = 2.1 nM T72335 C9UB1G 52949469 Ki = 90 nM T72335 CK2FC3 52949512 Ki = 1.3 nM T72335 CX61KT 52949570 Ki = 1 nM T72335 C47MHL 54579980 Ki = 1.5 nM T72335 CNC53R 54580455 Ki = 1.3 nM T72335 C6R3MZ 54580973 Ki = 1.2 nM T72335 CKEX38 54580974 Ki = 1.4 nM T72335 C2Z0ET 54581015 Ki = 0.36 nM T72335 CWKA42 54582019 Ki = 0.58 nM T72335 C27INL 54582020 Ki = 0.93 nM T72335 CXZ9K8 54582048 Ki = 0.25 nM T72335 C0ZE9W 54582049 Ki = 3.8 nM T72335 C86LQN 54582964 Ki = 0.81 nM T72335 C9N2LV 54582965 Ki = 0.68 nM T72335 C4V0KC 54582997 Ki = 1.1 nM T72335 CB5R3N 54582998 Ki = 1.2 nM T72335 CKMX69 54582999 Ki = 2 nM T72335 CA3WH5 54583957 Ki = 1.2 nM T72335 CU3LX7 54584000 Ki = 0.75 nM T72335 C7TO6F 54584001 Ki = 25 nM T72335 COS6J3 54584002 Ki = 5 nM T72335 CS93EQ 54585907 Ki = 577 nM T72335 C8SUM2 54586836 Ki = 4.6 nM T72335 CC5Q7W 54586877 Ki = 4.6 nM T72335 CXVL79 54586878 Ki = 3.1 nM T72335 C30TSN 54586879 Ki = 3.3 nM T72335 CHE2I1 57345500 Ki = 0.17 nM T72335 C63TFM 57345501 Ki = 0.31 nM T72335 C8KT2F 57345502 Ki = 0.27 nM T72335 C5JGB6 57393299 IC50 > 100000 nM T72335 C0NKX6 57393300 IC50 > 100000 nM T72335 CW8J0Q 57395004 IC50 > 100000 nM T72335 C8GAR4 57395030 IC50 > 100000 nM T72335 CRO42V 57396753 IC50 > 100000 nM T72335 C39RAT 57398522 IC50 > 100000 nM T72335 CA1MW7 57400217 IC50 > 100000 nM T72335 C8WN0U 57402018 IC50 > 100000 nM T72335 CE2BP6 57402019 IC50 > 100000 nM T72335 C1FAP4 59079459 IC50 > 100000 nM T72335 CVZN42 70683216 Ki = 0.23 nM T72335 C83VBO 70684920 IC50 = 1400 nM T72335 C7OTZ4 70684921 IC50 = 1700 nM T72335 C06KYR 70687076 IC50 > 10000 nM T72335 C6F3LR 70687441 Ki = 0.3 nM T72335 CVPQ62 70691618 Ki = 0.04 nM T72335 C7VZK0 70691619 Ki = 0.11 nM T72335 C2WF7D 70691628 Ki = 0.6 nM T72335 C1PL3K 70693705 Ki = 0.49 nM T72335 C0LVT8 70693709 Ki = 2 nM T72335 C6P3XM 70693710 Ki = 1 nM T72335 C51LCP 70695462 IC50 = 9500 nM T72335 CEX4A8 70695825 Ki = 1.3 nM T72335 CENQ98 70697478 IC50 = 2100 nM T72335 CTOQ24 73054451 IC50 = 70000 nM T72335 CTWG17 73054452 IC50 = 73000 nM T72335 CQI37A 73054453 IC50 > 100000 nM T72335 CUDC64 73054454 IC50 > 100000 nM T72335 CDHU61 73054455 IC50 > 100000 nM T72335 C79PZU 73054730 IC50 > 100000 nM T72335 CM9I1T 73054731 IC50 = 52000 nM T72335 CBV03K 73054732 IC50 = 81000 nM T72335 CN1R5T 73054733 IC50 = 90000 nM T72335 C9V6GC 73054734 IC50 = 44000 nM T72335 C63OXM 73054735 IC50 = 48000 nM T72335 CI14XA 73054736 IC50 = 43000 nM T72335 CK9TU0 73055013 Ki = 1140 nM T72335 CFPC79 73055014 IC50 = 17000 nM T72335 C1BY5E 73055015 IC50 = 55000 nM T72335 C7UQ1B 73055016 IC50 = 33000 nM T72335 CE86GN 73055017 IC50 > 100000 nM T72335 CO5FN4 73055018 Ki = 478 nM T72335 CMIN60 73055019 IC50 > 100000 nM T72335 C8EGU9 73055300 IC50 > 100000 nM T72335 C93ATJ 73055301 IC50 > 100000 nM T72335 CCK0B1 73055302 IC50 > 100000 nM T72335 CA9V7M 73055303 IC50 > 100000 nM T72335 CJ3VF9 73055304 IC50 > 100000 nM T72335 C3RFJ4 73055305 IC50 > 100000 nM T72335 CE3H7F 73055306 IC50 = 79000 nM T72335 CCX0B2 73055602 IC50 = 87000 nM T72335 C0E8XM 73055603 IC50 = 95000 nM T72335 C2AL5B 73055604 IC50 = 83000 nM T72335 C8H0UN 73055605 IC50 = 26000 nM T72335 CX80YH 73055606 IC50 = 61000 nM T72335 C80MBE 73055607 IC50 > 100000 nM T72335 C01SHT 73055902 IC50 = 3000 nM T72335 C2GE8Q 73055903 IC50 = 13000 nM T72335 CET0F1 73055904 IC50 = 10000 nM T72335 CDA75O 73055905 IC50 = 11000 nM T72335 CK5FT8 73055906 IC50 = 4600 nM T72335 C9OX6Y 73055907 IC50 = 5700 nM T72335 CA93JD 73056179 IC50 = 21000 nM T72335 CEX86T 73056180 IC50 = 33000 nM T72335 C8QZG6 73056181 IC50 = 36000 nM T72335 C9MK8R 73056182 IC50 > 100000 nM T72335 C1KGT9 73056183 IC50 = 38000 nM T72335 CB9PC2 73056184 IC50 > 100000 nM T72335 CR75BY 73056185 IC50 = 46000 nM T72335 CE5J8Z 73056473 IC50 > 100000 nM T72335 CW59QJ 73056474 IC50 > 100000 nM T72335 CSM32K 73056475 IC50 = 78000 nM T72335 CRB69T 73056476 IC50 = 58000 nM T72335 C67PCF 73056477 IC50 > 100000 nM T72335 C2ZPK9 73056478 IC50 > 100000 nM T72335 CVP2L3 73056479 IC50 > 100000 nM T72335 CDKP86 73056771 IC50 > 100000 nM T72335 C5TWA2 73056772 IC50 > 100000 nM T72335 C7YT0C 73056773 IC50 = 41000 nM T72335 C85VYZ 73056774 IC50 > 50000 nM T72335 C54NKF 73056775 IC50 > 100000 nM T72335 CU05BQ 92044070 IC50 = 9600 nM T72335 CIT0L9 122196479 IC50 = 7000 nM T72335 CW12YE 122196480 IC50 = 11000 nM T72335 CD78CQ 122196481 IC50 = 9500 nM T72335 C2WTM7 122196482 IC50 = 13000 nM T72335 CSUL01 122196483 IC50 = 14000 nM T72335 CK71TI 122196484 IC50 = 3400 nM T72335 CNW9L5 122196485 IC50 = 2100 nM T72335 CD14IW 122196486 IC50 = 3200 nM T72335 CNXM35 122196487 IC50 > 100000 nM T72335 C14KWN 122196488 IC50 = 29000 nM T72335 C98OTL 122196489 IC50 = 1700 nM T72335 CBM24K 122196490 IC50 = 1200 nM T72335 CA5U4V 122196492 IC50 = 1100 nM T72335 CK28UR 122196494 IC50 = 1300 nM T72335 CBI0Q8 122196496 IC50 = 1800 nM T72335 CE38OX 122196498 IC50 = 3700 nM T72335 CW7F9G 122196500 IC50 = 91000 nM T72335 CD63MB 122196501 IC50 = 16000 nM T72335 CRO6C1 122196502 IC50 = 15000 nM T72335 C04SMN 122196503 IC50 = 3200 nM T72335 C2FG3L 122196504 IC50 = 14000 nM T72335 CNH43Q 122196505 IC50 = 19000 nM T72335 C0DKI2 122196506 IC50 = 117000 nM T72335 CTYB74 122196507 IC50 = 9300 nM T72335 CT18AN 122196508 IC50 = 4800 nM T72335 CEG6I1 122196509 IC50 = 1300 nM T72335 C3B8XJ 135403140 Ki = 1100 nM T72335 C1LD6R 135457658 IC50 > 100000 nM T72335 C5RC3Z 136042247 IC50 > 100000 nM T72335 CH2NJ8 136042248 IC50 > 100000 nM T72335 C8KF9E 136042249 IC50 > 100000 nM T72335 CEF9L1 136043847 IC50 = 50000 nM T72335 CXTW67 136241621 IC50 = 14000 nM T72335 CWYJ60 137628929 IC50 = 199526.23 nM T72335 C07RUP 137629906 IC50 = 100000 nM T72335 C3EM4F 137631861 IC50 = 205 nM T72335 CW20RK 137633040 IC50 = 262 nM T72335 C1I2HL 137635814 IC50 = 197 nM T72335 CH01VT 137638628 IC50 = 83 nM T72335 C3K1CH 137641350 Ki = 18 nM T72335 C2TB0M 137645962 IC50 = 92 nM T72335 C61MRQ 137650294 IC50 = 1041 nM T72335 C04YGJ 137650967 IC50 = 6400 nM T72335 CP4SJ8 137654048 IC50 = 1942 nM T72335 C1LW5B 137654231 IC50 = 3500 nM T72335 CY5EZ4 137654626 IC50 = 250 nM T72335 CK6T4I 137654654 IC50 = 558 nM T72335 C3QD7K 137655213 IC50 = 61 nM T72335 CI85DX 137658315 IC50 = 221 nM T72335 C7OK2V 137658353 IC50 = 714 nM T72335 C9Q6CH 137658826 IC50 > 10000 nM T72335 CS9FT7 137661162 IC50 = 125 nM T72335 CQ2H4A 145964548 Ki = 946 nM T72335 C0EXI5 145964588 EC50 = 60 nM T72335 CTHV30 145966256 IC50 > 10000 nM T72335 CI8G5Z 145966625 Ki = 946 nM T72335 C0GKU1 145968929 EC50 = 104.6 nM T72335 CNX3J8 145968930 EC50 = 12 nM T72335 CW5OJ9 145973096 EC50 = 23.7 nM T72335 CS14PQ 145975108 EC50 = 31.7 nM T72335 CNMD49 145976619 Ki = 1173 nM T72335 D01QWL 44454145 Ki = 2200 nM T72335 D03QAN 71166 Ki = 500 nM T72335 D0A4TC 446504 IC50 = 1200 nM T72335 D0EL3A 44454442 Ki = 6200 nM T72335 D0I1NU 72392 Ki = 42900 nM T72335 D0J5VK 67145 Ki = 2400 nM T72335 D0M2KQ 23661707 Ki = 1700 nM T72335 D0M4IF 5282106 Ki = 3000 nM T72335 D0M9DT 5282309 IC50 = 2300 nM T72335 D0MV0W 1138119 IC50 = 3000 nM T72335 D0SU7B 44441632 Ki = 6000 nM T72335 D0TO6S 2396 IC50 = 1500 nM T72335 D0X1JG 213329 IC50 = 15000 nM T62391 D00ENY 33032 EC50 = 3660 nM T62391 D03CNS 2910 EC50 = 13700 nM T62391 D02VKC 3272524 Ki = 900 nM T62391 D0B0NQ 127894 Ki = 32000 nM T62391 COC91V 10255 EC50 = 26610 nM T62391 CC0E1V 447081 Ki = 2.24 nM T62391 CNBI79 447083 EC50 = 1600 nM T62391 CO28NU 447407 EC50 = 7900 nM T62391 C1EP3D 2733518 Ki = 12000 nM T62391 CWK7X4 4694356 Ki = 27500 nM T62391 C3JXD9 5289518 EC50 = 32000 nM T62391 C9TLQ4 9861035 Ki > 10000 nM T62391 CFV03Y 9926589 Ki = 247000 nM T62391 CFC2P8 9928016 EC50 = 1660 nM T62391 C7Q1MJ 10132082 IC50 > 100000 nM T62391 CFKJ76 10352480 Ki = 160 nM T62391 C1N2VM 10420002 Ki = 1070 nM T62391 C0O6ZI 10658567 EC50 > 3000000 nM T62391 CQ38WM 11219775 Ki = 1180 nM T62391 CGRT02 11288627 Ki = 44.8 nM T62391 CHUX80 11818375 Ki = 3710 nM T62391 CQ2YP8 16659202 EC50 = 1000000 nM T62391 CDZ2E6 18713992 EC50 = 1660 nM T62391 C38HPQ 46886654 EC50 = 41600 nM T62391 C56NLW 127039193 EC50 > 1000000 nM T62391 C5Q6ZI 137638800 Ki = 13900 nM T62391 C03KAU 155519563 EC50 > 1000000 nM T62391 D03RGP 1221 Ki = 21 nM T62391 D09LXQ 126569 EC50 = 20900 nM T62391 D0KD6O 5288598 EC50 = 7200 nM T62391 D0N1CL 9799478 IC50 > 100000 nM T62391 D0O7OE 122294 IC50 = 230 nM T62391 D0SB9H 119582 IC50 = 30 nM T62391 D0T5SU 158397 Ki = 20.6 nM T24793 D04OSE 4485 IC50 = 1350 nM T24793 D0G7HO 9905818 IC50 = 32000 nM T24793 C7DAX1 10338800 IC50 = 12200 nM T24793 CY0EX6 10914479 IC50 = 2800 nM T24793 C02HTI 14532695 IC50 = 24000 nM T24793 C91QFN 25019282 IC50 = 23400 nM T24793 CSE6Z5 71463101 EC50 > 100000 nM T24793 CY9J7D 90656507 IC50 = 18700 nM T24793 CY07BI 90656508 IC50 = 12800 nM T24793 C9OH0X 90656509 IC50 = 9900 nM T24793 C17FMR 90656510 IC50 = 95800 nM T24793 C2GZ9H 90656511 IC50 = 27100 nM T24793 CI42MU 90656512 IC50 = 9300 nM T24793 C7X0BY 90656513 IC50 = 28400 nM T24793 C0Z4AG 90656514 IC50 = 29800 nM T24793 CE1YH5 90656515 IC50 = 26800 nM T24793 C2E4CW 90656516 IC50 = 15100 nM T24793 CEX5V3 90656517 IC50 = 59600 nM T24793 CLA3B5 90656518 IC50 = 56200 nM T24793 CYW8C7 90656519 IC50 > 100000 nM T24793 C82HOY 90656520 IC50 = 20600 nM T24793 C1QT6R 90656521 IC50 = 18500 nM T24793 C7A2KQ 90656522 IC50 = 44100 nM T24793 CP08NQ 90656523 IC50 = 57100 nM T24793 CIB1Z0 90656524 IC50 = 14900 nM T24793 CK0O4F 90656525 IC50 = 55500 nM T24793 CA3I1P 90656526 IC50 = 63100 nM T57034 CG48YC 97710 IC50 = 139000 nM T57034 CGO87D 109515 IC50 = 3900 nM T57034 CQ4C2L 236027 Ki = 73200 nM T57034 CONR62 444765 Ki = 11000 nM T57034 C9B3YM 444766 Ki = 560000 nM T57034 CM0IQ3 446665 IC50 = 342000 nM T57034 C5Y3DJ 446871 Ki = 21000 nM T57034 CAR67L 457943 IC50 = 31000 nM T57034 CE3S9R 1820399 IC50 = 59400 nM T57034 C35LZP 4774445 Ki = 19000 nM T57034 CL5IF1 5179836 IC50 = 135000 nM T57034 CPM09B 5327156 IC50 = 20700 nM T57034 CJ0AT8 5383687 Ki = 26000 nM T57034 CF48XG 6914659 Ki = 200 nM T57034 C4BE0F 9874843 IC50 = 500 nM T57034 CA75NG 9985013 IC50 = 77000 nM T57034 C3A8JL 10256983 IC50 = 15000 nM T57034 CZTN01 10675368 IC50 = 600 nM T57034 CT4H0O 11006141 IC50 = 77000 nM T57034 C2WP1J 11343454 IC50 = 32000 nM T57034 COIR53 11456678 IC50 = 13000 nM T57034 CYE98M 14295338 IC50 = 3800 nM T57034 CBJ60K 18864315 IC50 = 400 nM T57034 CWU92E 20866464 IC50 > 50000 nM T57034 CJKO23 20866499 IC50 = 14400 nM T57034 C1OR3D 22084082 Ki = 3600 nM T57034 C5O0SV 24204784 IC50 = 100 nM T57034 CZL2T6 24815971 IC50 = 0.3 nM T57034 CT20HY 44359237 Ki = 18000 nM T57034 C5YV1R 44359299 Ki = 160000 nM T57034 C4Z6WR 44434444 IC50 = 1100 nM T57034 C2VU4R 44585540 Ki = 220 nM T57034 CJX8B4 45379330 IC50 = 130 nM T57034 C1ULD8 45483667 Ki = 14000 nM T57034 C45AFN 46186815 Ki > 100000 nM T57034 C2IU1Z 49796692 IC50 = 300000 nM T57034 C8OM7T 49797143 IC50 = 430 nM T57034 CXP8Q1 49797144 IC50 = 300 nM T57034 C7DR6K 49797145 IC50 = 410 nM T57034 CCNW45 49797146 IC50 = 290 nM T57034 CSYI82 49797147 IC50 = 140 nM T57034 C3N4WV 49797148 IC50 = 150 nM T57034 C8B5IL 49797149 IC50 = 380 nM T57034 C3Z9XK 49797150 IC50 = 90 nM T57034 C6LN5C 49797153 IC50 = 230 nM T57034 C7YPR2 49797154 IC50 = 230 nM T57034 C4NYB5 49797155 IC50 = 570 nM T57034 CZR0Y3 49797156 IC50 = 150 nM T57034 C0E5MB 49797157 IC50 = 270 nM T57034 C6OE0U 49797158 IC50 = 200 nM T57034 CXQ18O 49797159 IC50 = 80 nM T57034 CRJ69K 49797160 IC50 = 420 nM T57034 C3Y0IQ 49797161 IC50 = 390 nM T57034 C0PZ7R 49797162 IC50 = 330 nM T57034 CH6W8N 49797163 IC50 = 60 nM T57034 C51LVT 49797164 IC50 = 100 nM T57034 C64QPY 49797165 IC50 = 80 nM T57034 C0QH5S 49797166 IC50 = 1000 nM T57034 CTY7U4 49797167 IC50 = 450 nM T57034 C9YZ7F 49797168 IC50 = 70 nM T57034 C4V3AU 49797169 IC50 = 400 nM T57034 C9FZU2 49797170 IC50 = 340 nM T57034 C3T9BD 49797171 IC50 = 210 nM T57034 C27QAD 52941367 IC50 = 4500 nM T57034 CU5ND3 57514697 IC50 > 200000 nM T57034 C2BT9H 70673568 IC50 = 12000 nM T57034 CCY15D 71734765 IC50 = 470 nM T57034 CMC9L2 72190151 IC50 = 18000 nM T57034 CM1W6X 73352369 IC50 = 12000 nM T57034 C12OHP 122187565 IC50 > 50000 nM T57034 CXHR32 122187566 IC50 > 50000 nM T57034 C59OUG 122187567 IC50 > 50000 nM T57034 D0E0BU 444763 Ki = 6000 nM T57034 D0Y1RO 1829 Ki = 17000 nM T57034 D0Y5SB 444764 Ki = 33000 nM T68706 CSM4Q6 262935 Ki = 376000 nM T68706 COFC54 5347695 Ki = 11800 nM T68706 C0FJG2 5916478 Ki = 273000 nM T68706 C62WJS 6332610 Ki = 44000 nM T68706 CP3QT1 9560223 Ki = 1470 nM T68706 C9QW6K 9568045 Ki > 500000 nM T68706 C7XL2M 9573034 Ki = 1840 nM T68706 C25WST 9573756 Ki = 17300 nM T68706 CMKZ82 9574209 Ki = 4780 nM T68706 CGT32J 9994348 Ki = 1820 nM T68706 CED36V 10009347 Ki = 6400 nM T68706 C16CXQ 10033400 Ki = 900 nM T68706 CJ5CA8 10105958 Ki = 11500 nM T68706 C8OC6J 10212767 Ki = 990 nM T68706 C4C5AF 10219094 Ki = 420 nM T68706 C75TFE 10259947 Ki = 1900 nM T68706 CC46LA 10485685 Ki = 190 nM T68706 CBUF92 11228390 Ki = 1.7 nM T68706 CUIM84 11628682 Ki = 169 nM T68706 CZ78TN 11650945 Ki = 114 nM T68706 CFHX82 11837140 IC50 > 50000 nM T68706 C3RV5A 16043267 Ki = 6 nM T68706 CK7Y2E 16757513 Ki = 23 nM T68706 CL2K9U 20333093 IC50 > 50000 nM T68706 C2T4QJ 25195678 Ki = 138 nM T68706 CW1A4N 25196726 IC50 > 50000 nM T68706 C2FU9P 42618077 IC50 > 50000 nM T68706 CWXJ06 44156975 IC50 > 50000 nM T68706 C58KSV 44156976 IC50 > 50000 nM T68706 C4EZF0 44352560 Ki = 240 nM T68706 CK5HB4 44352627 Ki = 350 nM T68706 CK9BD0 44352629 Ki = 5.1 nM T68706 C0CFN6 44352635 Ki = 3.4 nM T68706 C97MNE 44352636 Ki = 7.5 nM T68706 CY4OG7 44352637 Ki = 370 nM T68706 C58IZU 44352651 Ki = 26 nM T68706 C4Z7EM 44352695 Ki = 330 nM T68706 CT3Q5N 44584806 Ki = 67 nM T68706 C5A9HE 44584807 Ki > 100 nM T68706 CJ0X2K 44584808 Ki > 100 nM T68706 CK73GW 44584809 Ki > 100 nM T68706 CI81BN 44584810 Ki > 100 nM T68706 C41POU 44584811 Ki > 100 nM T68706 C61OSN 44584812 Ki = 57 nM T68706 CB6Y4T 44584813 Ki > 100 nM T68706 CG1L4I 44584814 Ki > 100 nM T68706 CR0S1A 44584815 Ki > 100 nM T68706 CW4DN7 44584816 Ki > 100 nM T68706 CLW5C3 44584817 Ki > 100 nM T68706 CSB8X3 44584818 Ki > 100 nM T68706 CCTP19 44584819 Ki > 100 nM T68706 C29EYG 44584820 Ki > 100 nM T68706 CFR2M3 44584821 Ki > 100 nM T68706 CKG1U6 44584822 Ki > 100 nM T68706 C62FAQ 44584823 Ki > 100 nM T68706 C2K8OA 44584824 Ki > 100 nM T68706 CUF8E5 44584825 Ki > 100 nM T68706 C0X4KU 44584826 Ki > 100 nM T68706 COE8L9 44584827 Ki > 100 nM T68706 CG0KU3 44584828 Ki > 100 nM T68706 CY3V8P 44584829 Ki > 100 nM T68706 CD6ZC5 44584830 Ki > 100 nM T68706 C9UN5P 44584831 Ki > 100 nM T68706 CA0DC8 44584832 Ki > 100 nM T68706 CS27KE 44584833 Ki > 100 nM T68706 CFN4J7 44584834 Ki > 100 nM T68706 C65LUD 44584835 Ki > 100 nM T68706 CUX56H 44584836 Ki > 100 nM T68706 CS98BC 44584837 Ki > 100 nM T68706 C27ROJ 44584838 Ki > 100 nM T68706 CIB62U 44584839 Ki > 100 nM T68706 CBWC20 44584840 Ki > 100 nM T68706 CRQK05 44584841 Ki > 100 nM T68706 CT37IE 44584842 Ki > 100 nM T68706 CPL2H1 44584843 Ki > 100 nM T68706 CM29XN 44584844 Ki = 80 nM T68706 C32LWT 44584845 Ki > 100 nM T68706 CUS16Z 44584846 Ki = 30 nM T68706 CB5F0T 44584847 Ki > 100 nM T68706 CD58FL 44584848 Ki = 38 nM T68706 C3PN7C 44584849 Ki = 59 nM T68706 CQE24W 44584850 Ki > 100 nM T68706 CUQ9K4 44584863 Ki > 100 nM T68706 CE3MW2 44584948 Ki > 100 nM T68706 CQH8U7 44584950 Ki = 45 nM T68706 CPYT15 44584951 Ki = 47 nM T68706 CUZ71D 44584952 Ki = 56 nM T68706 CP2J8X 44584953 Ki = 33 nM T68706 CJKB12 44584954 Ki > 100 nM T68706 CF3Y6V 44584955 Ki > 100 nM T68706 C73YFH 44584956 Ki > 100 nM T68706 CMD1Z7 44584957 Ki > 100 nM T68706 CAOR08 44584958 Ki = 65 nM T68706 CF2LH5 44584959 Ki = 81 nM T68706 CBX8K0 44584960 Ki = 34 nM T68706 C10KCB 44584961 Ki = 38 nM T68706 C1S6KQ 44584962 Ki = 47 nM T68706 CDCH27 44584964 Ki > 100 nM T68706 C31PGM 44584965 Ki > 100 nM T68706 CQOC14 44584966 Ki > 100 nM T68706 C0GF2Q 44584967 Ki > 100 nM T68706 CF7KY4 44584968 Ki > 100 nM T68706 C4LHQ9 44584969 Ki > 100 nM T68706 C9X3FD 44584970 Ki > 100 nM T68706 CQSO90 44584971 Ki > 100 nM T68706 CD37QK 44584972 Ki > 100 nM T68706 C0G3MD 44584973 Ki > 100 nM T68706 CJM03L 44584974 Ki > 100 nM T68706 CT47PD 44584975 Ki > 100 nM T68706 CJ1P5B 44584976 Ki > 100 nM T68706 CEMD30 44584977 Ki > 100 nM T68706 CD71WT 44584978 Ki > 100 nM T68706 CG2KE0 44584979 Ki > 100 nM T68706 CLC8K5 44584980 Ki > 100 nM T68706 CF9RK1 44584981 Ki > 100 nM T68706 C9CEO7 44584982 Ki > 100 nM T68706 CXNK25 44584983 Ki > 100 nM T68706 CNA4O5 44584984 Ki > 100 nM T68706 C1J0LO 44584985 Ki > 100 nM T68706 C67DIC 44584986 Ki > 100 nM T68706 CX79JW 44584987 Ki > 100 nM T68706 CKM6J1 44584988 Ki > 100 nM T68706 C9OX8T 44584989 Ki > 100 nM T68706 CQP51O 44584990 Ki > 100 nM T68706 CP7KN4 44584991 Ki > 100 nM T68706 CJXP53 44584992 Ki > 100 nM T68706 CEB46O 44584993 Ki > 100 nM T68706 CNC7Y0 44584994 Ki > 100 nM T68706 CS02PI 44584995 Ki > 100 nM T68706 CB2K4M 44584996 Ki > 100 nM T68706 C3FE4S 44584997 Ki > 100 nM T68706 C8MAW2 44584998 Ki > 100 nM T68706 CNB4L3 44584999 Ki > 100 nM T68706 CXL76H 44585000 Ki > 100 nM T68706 C47OBC 44585001 Ki > 100 nM T68706 C3JYM7 44585002 Ki > 100 nM T68706 CG71FH 44585004 Ki > 100 nM T68706 C4CSQ2 44585005 Ki > 100 nM T68706 C7ZO5P 44585006 Ki > 100 nM T68706 CK5VW7 44585007 Ki > 100 nM T68706 CG0OR5 44585008 Ki > 100 nM T68706 C78MRO 44585009 Ki > 100 nM T68706 CR27AE 44585010 Ki > 100 nM T68706 C8M7DI 44585011 Ki > 100 nM T68706 COEC52 44585012 Ki > 100 nM T68706 CKG8S2 44585013 Ki > 100 nM T68706 CST23K 44585014 Ki > 100 nM T68706 C4BSZ6 44585015 Ki > 100 nM T68706 CO1E8Z 44585016 Ki > 100 nM T68706 C5KJ9Q 44585017 Ki > 100 nM T68706 CQX41M 44585018 Ki > 100 nM T68706 CI6AW8 44585019 Ki > 100 nM T68706 C34MRQ 44585020 Ki > 100 nM T68706 CNQR65 44585021 Ki > 100 nM T68706 C8Z4WQ 44585022 Ki > 100 nM T68706 CWEI08 44585023 Ki > 100 nM T68706 C1UF2C 44585024 Ki > 100 nM T68706 C32TRO 44585025 Ki > 100 nM T68706 CU9CH7 44585026 Ki > 100 nM T68706 C5WVR1 44585027 Ki > 100 nM T68706 CC4P1B 44585028 Ki > 100 nM T68706 C4ZQP1 44585029 Ki > 100 nM T68706 CGML74 44585030 Ki > 100 nM T68706 C8SM9K 44585031 Ki > 100 nM T68706 CWC2Y9 44585032 Ki > 100 nM T68706 CZH7M3 44585033 Ki > 100 nM T68706 CZ7S2E 44585034 Ki > 100 nM T68706 CG60WN 44585035 Ki > 100 nM T68706 CMV32T 44585036 Ki > 100 nM T68706 CN74EF 44585037 Ki > 100 nM T68706 CCTM89 44585038 Ki > 100 nM T68706 CC25VQ 44585039 Ki > 100 nM T68706 CY3CG4 44585040 Ki > 100 nM T68706 CV1F3G 44585041 Ki > 100 nM T68706 C8KOE2 44585042 Ki > 100 nM T68706 CG9CO3 44585043 Ki > 100 nM T68706 CZ9F8X 44585044 Ki = 115 nM T68706 CC8MJ0 44585045 Ki = 48 nM T68706 C9MR4W 44585046 Ki > 100 nM T68706 CB7N5J 44585047 Ki > 100 nM T68706 CH7C1E 44585048 Ki > 100 nM T68706 CG0UK7 44585049 Ki = 103 nM T68706 C7PYW8 44585050 Ki > 100 nM T68706 C5JHS4 44585051 Ki = 58 nM T68706 C1PDB6 44585052 Ki > 100 nM T68706 CL9PD0 44585053 Ki > 100 nM T68706 CC0V7O 44585054 Ki > 100 nM T68706 C8UBS3 44585055 Ki > 100 nM T68706 CA1PS3 44585056 Ki = 50 nM T68706 CE2PV8 44585057 Ki > 100 nM T68706 CBM2Y7 44585058 Ki > 100 nM T68706 CZVN12 44585059 Ki > 100 nM T68706 C7T3LQ 44585060 Ki > 100 nM T68706 CKH27O 44585061 Ki > 100 nM T68706 CAZ34N 44585062 Ki = 93 nM T68706 C4VD2W 44585063 Ki > 100 nM T68706 CQV2W1 44585064 Ki > 100 nM T68706 C3YJL1 44585065 Ki > 100 nM T68706 CGA7K6 44585066 Ki > 100 nM T68706 CLBV32 44585067 Ki > 100 nM T68706 CQIJ72 44585068 Ki > 100 nM T68706 CG02SN 44585069 Ki > 100 nM T68706 C98HFK 44585070 Ki > 100 nM T68706 C9T5CZ 44585071 Ki > 100 nM T68706 CRL9H6 44585072 Ki > 100 nM T68706 CHA0M1 44585073 Ki > 100 nM T68706 C1F3XD 44585074 Ki > 100 nM T68706 C82EPA 44585075 Ki > 100 nM T68706 CGX5C2 44585076 Ki > 100 nM T68706 CF8B5L 44585077 Ki > 100 nM T68706 CP7K4R 44585078 Ki > 100 nM T68706 CT2MV6 44585079 Ki > 100 nM T68706 C1R9XI 44585080 Ki > 100 nM T68706 CXC08A 44585081 Ki > 100 nM T68706 CLC7S0 44585082 Ki > 100 nM T68706 C0QH7B 44585083 Ki > 100 nM T68706 CX70KM 44585084 Ki > 100 nM T68706 CO0N2T 44585085 Ki > 100 nM T68706 C42TGS 44585086 Ki > 100 nM T68706 C58ZDW 44585087 Ki > 100 nM T68706 C45NBG 44585088 Ki > 100 nM T68706 CVD73E 44585089 Ki > 100 nM T68706 C49VDL 44585090 Ki > 100 nM T68706 CC61AT 44585091 Ki > 100 nM T68706 C2F8QP 44585092 Ki > 100 nM T68706 CIP31K 44585093 Ki > 100 nM T68706 COJ28W 44585094 Ki > 100 nM T68706 C9RGX0 44585095 Ki > 100 nM T68706 C4ZUP3 44585096 Ki > 100 nM T68706 C06VHK 44585097 Ki > 100 nM T68706 CPJ9K4 44585099 Ki > 100 nM T68706 CWT6A4 44585100 Ki > 100 nM T68706 C9MWI6 44585101 Ki > 100 nM T68706 CNZ81Q 44585102 Ki = 39 nM T68706 CE4WN9 44585107 Ki = 42 nM T68706 C6X1HU 44585113 Ki > 100 nM T68706 C8X1KW 44585114 Ki > 100 nM T68706 CU5KY2 44585115 Ki > 100 nM T68706 CU27NO 44585116 Ki > 100 nM T68706 CGK50M 44585117 Ki > 100 nM T68706 CQD4Z8 44585118 Ki > 100 nM T68706 C94ZCT 44585119 Ki = 57 nM T68706 C2ZWE4 44585120 Ki > 100 nM T68706 CK7XM0 44585121 Ki > 100 nM T68706 CN3AD9 44585122 Ki > 100 nM T68706 C7RI5O 44585123 Ki > 100 nM T68706 C0ZBN3 44585124 Ki > 100 nM T68706 CC75XO 44585125 Ki > 100 nM T68706 CWNB15 44585126 Ki > 100 nM T68706 C57HGE 44585127 Ki = 80 nM T68706 CI09DY 44585128 Ki > 100 nM T68706 CJ7LF5 44585129 Ki = 30 nM T68706 CO93HF 44585130 Ki = 38 nM T68706 C0MJN2 44585131 Ki > 100 nM T68706 C8V5GT 44585132 Ki = 59 nM T68706 CIRV70 44585133 Ki > 100 nM T68706 C2RNK5 44585134 Ki > 100 nM T68706 CRW3B9 44585135 Ki > 100 nM T68706 CVTE96 44585136 Ki = 53 nM T68706 C2W5AH 44585137 Ki = 45 nM T68706 C9TFD6 44585138 Ki = 47 nM T68706 C7X2UH 44585139 Ki = 56 nM T68706 C1H2WG 44585140 Ki > 100 nM T68706 CRL0A6 44585141 Ki > 100 nM T68706 CT1N4A 44585142 Ki > 100 nM T68706 CZ6SO5 44585143 Ki > 100 nM T68706 CG8R2Y 44585144 Ki = 65 nM T68706 CS4TQ6 44585145 Ki = 81 nM T68706 CO56MF 44585146 Ki > 100 nM T68706 C9SW4V 44585147 Ki > 100 nM T68706 C46BYS 44585148 Ki > 100 nM T68706 CIJ0Z8 44585149 Ki > 100 nM T68706 C79UBQ 44585150 Ki > 100 nM T68706 C8YO5T 44585151 Ki > 100 nM T68706 CW5A2K 44585152 Ki > 100 nM T68706 C56DTX 44585153 Ki > 100 nM T68706 CFDC58 44585154 Ki > 100 nM T68706 CVL28O 44585155 Ki > 100 nM T68706 C6C4MS 44585156 Ki > 100 nM T68706 C4C7HG 44585157 Ki > 100 nM T68706 CDI21X 44585158 Ki > 100 nM T68706 CKIJ08 44585159 Ki > 100 nM T68706 C8R5YX 44585160 Ki > 100 nM T68706 CYC8R9 44585161 Ki > 100 nM T68706 CCRD92 44585162 Ki > 100 nM T68706 CJV7X2 44585163 Ki > 100 nM T68706 C5TDU2 44585164 Ki > 100 nM T68706 CQFC87 44585165 Ki > 100 nM T68706 CUA85D 44593129 Ki = 89 nM T68706 C7P8EK 44593130 Ki = 404 nM T68706 C4JS9X 44593146 Ki = 22 nM T68706 CQ4OK8 44593147 Ki = 69 nM T68706 C20JPC 44593148 Ki = 12 nM T68706 CUZ62D 44593168 Ki = 42 nM T68706 C6S5JH 44593169 Ki = 46 nM T68706 CNT7J8 44593170 Ki = 423 nM T68706 C0Q9CE 44593171 Ki = 812 nM T68706 CWP01R 44593172 Ki = 1768 nM T68706 CV07SM 44593173 Ki = 100000 nM T68706 CEW2O5 44593174 Ki = 100000 nM T68706 CB80ER 44593175 Ki = 100000 nM T68706 CE3CR0 44593197 Ki = 100000 nM T68706 C2YPS6 44593198 Ki = 100000 nM T68706 C7P5LR 44593199 Ki = 100000 nM T68706 CN3EB5 44612015 Ki = 800 nM T68706 CGF70P 45486343 Ki = 3020 nM T68706 CNOP07 45486344 Ki = 63 nM T68706 C4G3BC 45486345 Ki = 7490 nM T68706 CJ73BT 45486346 Ki = 78 nM T68706 CF9I7Y 45486347 Ki = 553 nM T68706 C1NIR6 45486348 Ki = 1070 nM T68706 CAJQ48 45486349 Ki = 627 nM T68706 C6EB3A 45486350 Ki = 1430 nM T68706 CW8RA2 45486351 Ki = 1320 nM T68706 CQS4W0 45486352 Ki = 2730 nM T68706 CSX01I 45486353 Ki = 9710 nM T68706 C9ETC4 45486354 Ki = 53 nM T68706 CVPG40 45486356 Ki = 1.6 nM T68706 CSQ2K4 45486357 Ki = 1 nM T68706 CL4D9S 45486358 Ki = 3.3 nM T68706 CDE58N 46191000 Ki = 285 nM T68706 CAJL68 46191001 Ki = 702 nM T68706 CG1HV0 46191002 Ki = 1.5 nM T68706 C8FP5E 46191072 Ki = 7340 nM T68706 C7NM3V 46191073 Ki = 37 nM T68706 C3X0OE 46191074 Ki = 24 nM T68706 CWL5Q8 46191148 Ki = 6 nM T68706 C5YX7K 46191149 Ki = 3 nM T68706 C8Z6SQ 46191150 Ki = 3.7 nM T68706 CYN8K9 46191291 Ki = 40 nM T68706 C9NC7I 46191292 Ki = 19 nM T68706 C2INC9 46191293 Ki = 3 nM T68706 CR7I8G 46191363 Ki = 3.6 nM T68706 CV1X4F 46191364 Ki = 1.4 nM T68706 CT26LP 46191365 Ki = 0.84 nM T68706 CQGL01 46191433 Ki = 12 nM T68706 CQ1MA3 46191434 Ki = 6.3 nM T68706 C32SJP 46191435 Ki = 23 nM T68706 C97QIZ 46191505 Ki = 405 nM T68706 CJZA45 46232267 IC50 > 50000 nM T68706 C3PLE6 46232269 IC50 > 50000 nM T68706 C3U8HV 46232270 IC50 > 50000 nM T68706 CYA73D 46232312 IC50 > 50000 nM T68706 C9Q7YX 53317374 Ki = 27900 nM T68706 CA86OS 53317375 Ki = 1130 nM T68706 C93QWB 53318957 Ki = 5610 nM T68706 C4W1DB 53320248 Ki = 1130 nM T68706 CLO86W 53321180 Ki = 580 nM T68706 CGZC91 53321290 Ki = 173000 nM T68706 C7QEI1 53321291 Ki = 460 nM T68706 CFOI53 53322612 Ki = 1550 nM T68706 CWA7B3 53323948 Ki = 1040 nM T68706 CSYV84 53325117 Ki = 1940 nM T68706 CQ7D3S 53325118 Ki = 1350 nM T68706 CO6TG4 53325236 Ki = 1420 nM T68706 CO0R2M 53325237 Ki = 1200 nM T68706 C8G4SM 53326426 Ki = 1460 nM T68706 CSP13L 53380708 Ki = 0.83 nM T68706 C2NYC4 53380709 Ki = 1.9 nM T68706 CB2W7R 56660089 Ki = 13 nM T68706 CTN23H 56660090 Ki = 1110 nM T68706 CCG0B8 56660091 Ki = 2390 nM T68706 CD1X9B 56663556 Ki = 3200 nM T68706 C9P3SV 56667001 Ki = 5.9 nM T68706 C6K5AI 56670442 Ki = 970 nM T68706 CX3F7D 56673930 Ki = 102 nM T68706 CVA9L6 56673931 Ki = 238 nM T68706 CY28PE 56673932 Ki = 1385 nM T68706 C2GXS8 56677267 Ki = 9.7 nM T68706 CEPU28 56680566 Ki = 142 nM T68706 CV3H4S 56683904 Ki = 6.3 nM T68706 C8ON3V 70684173 Ki = 3020 nM T68706 C4O8IR 70684174 Ki = 7490 nM T68706 CF78WO 70684175 Ki = 1070 nM T68706 CU9BW3 70684182 Ki = 2730 nM T68706 CGX63U 70684183 Ki = 3500 nM T68706 CYK60H 70686317 Ki = 1 nM T68706 C0TCG9 70686318 Ki = 3.3 nM T68706 C2XUM9 70686319 Ki = 3400 nM T68706 C4ESI6 70688429 Ki = 1.6 nM T68706 C87OHL 70690464 Ki = 63 nM T68706 C3R9EA 70690465 Ki = 78 nM T68706 C2MD9T 70690466 Ki = 1320 nM T68706 CUCP34 70690475 Ki = 53 nM T68706 CA9YT3 70692619 Ki = 1430 nM T68706 C9MVW4 70694663 Ki = 553 nM T68706 C41VFE 70694672 Ki = 9710 nM T68706 CDEV58 70694673 Ki = 0.81 nM T68706 CG4C9F 70696704 Ki = 627 nM T68706 C6TO1L 71450124 Ki = 1000 nM T68706 C8F5YQ 71451941 Ki > 1000 nM T68706 CGD6J4 71451942 Ki = 400 nM T68706 CY86ZW 71453763 Ki = 1300 nM T68706 C5I3EB 71453792 Ki = 500 nM T68706 CT51YJ 71453793 Ki = 1.4 nM T68706 C7WM6Z 71455497 Ki = 430 nM T68706 C35YRK 71457282 Ki = 2600 nM T68706 C2YEU4 71457318 Ki = 760 nM T68706 CB9MG1 71459125 Ki = 12.4 nM T68706 C0N8UR 71460934 Ki = 2.9 nM T68706 CDLP98 71460935 Ki = 5.3 nM T68706 CIS3R0 71460936 Ki = 4100 nM T68706 CK1X0W 71462644 Ki = 9 nM T68706 CGR35S 71462645 Ki = 1200 nM T68706 CQNG13 71608634 Ki = 9.8 nM T68706 C6HAL4 73345659 Ki > 100 nM T68706 CK7O6Q 73350255 Ki = 53 nM T68706 C4APW2 75593416 Ki = 680 nM T68706 CJ2W9V 75593418 Ki = 27 nM T68706 C29QOJ 76310654 Ki = 980 nM T68706 CAT6S5 76310655 Ki = 9550 nM T68706 CG87ZE 76310656 Ki = 7300 nM T68706 CQ7TE3 76310980 Ki = 8 nM T68706 CV8Z5G 76314290 Ki = 800 nM T68706 CULA07 76314608 Ki = 89 nM T68706 C6BT0I 76314609 Ki = 6 nM T68706 C6ZXN7 76314610 Ki = 1.9 nM T68706 CGB4J9 76317836 Ki = 650 nM T68706 C7G4XB 76317837 Ki = 560 nM T68706 CFXK67 76317855 Ki = 950 nM T68706 C6JAY9 76318181 Ki = 123 nM T68706 CYJ1I9 76318182 Ki = 21 nM T68706 CH3N0A 76321557 Ki = 1980 nM T68706 CF78UP 76321572 Ki = 1070 nM T68706 CX5I2O 76321887 Ki = 18 nM T68706 CA5K8R 76321888 Ki = 591 nM T68706 CMYK97 76325157 Ki = 980 nM T68706 CZ62KS 76328735 Ki = 2300 nM T68706 C4LG2O 76328736 Ki = 2100 nM T68706 C2J7OP 76329062 Ki = 25 nM T68706 CDC1J5 76329063 Ki = 33 nM T68706 CIY15Q 76332398 Ki = 2550 nM T68706 CL2ZX3 76332418 Ki = 2800 nM T68706 CX2VL4 76336024 Ki = 1120 nM T68706 CGZN04 76336044 Ki = 11000 nM T68706 C0ET8W 137630787 Ki = 1 nM T68706 CC3V7S 137631353 Ki = 3 nM T68706 C2JV6R 137631479 Ki = 0.4 nM T68706 C53MJF 137631755 Ki = 3 nM T68706 CN26ME 137631991 Ki = 11.7 nM T68706 CUOC87 137632800 Ki = 2 nM T68706 C5VFZ9 137633317 Ki = 3.1 nM T68706 C73DJB 137633620 Ki = 5 nM T68706 CBNJ52 137633770 Ki = 5.9 nM T68706 CRN21S 137633930 Ki = 50 nM T68706 CP8DN5 137634404 Ki = 0.9 nM T68706 CAIC85 137634503 Ki = 3 nM T68706 C0T3NR 137635077 Ki = 5 nM T68706 C9MUE6 137636542 Ki = 4.5 nM T68706 CG95RB 137636600 Ki = 4 nM T68706 C4GHK8 137636619 Ki = 4 nM T68706 CG5Q8T 137636730 Ki = 1.7 nM T68706 CH8AU1 137636950 Ki = 13 nM T68706 CDVJ93 137637528 Ki = 18 nM T68706 C5DX1A 137637600 Ki = 2.3 nM T68706 CDY46K 137637620 Ki = 260 nM T68706 C87STU 137638937 Ki = 30 nM T68706 C5L0NC 137639050 Ki = 4 nM T68706 CBH65X 137639397 Ki = 12 nM T68706 CN0FY7 137639688 Ki = 0.5 nM T68706 CJMG20 137640300 Ki = 13 nM T68706 CB2Z9N 137640311 Ki = 4 nM T68706 CERC30 137640559 Ki = 1.8 nM T68706 C35AYG 137641095 Ki = 3 nM T68706 CUM15D 137641134 Ki = 140 nM T68706 CQ76RK 137641874 Ki = 6 nM T68706 CO3S8F 137641997 Ki = 6 nM T68706 CMA50S 137642172 Ki = 0.5 nM T68706 C5AM0F 137642389 Ki = 5 nM T68706 CNC1O3 137642533 Ki = 36 nM T68706 CA5PJ2 137642642 Ki = 2.6 nM T68706 CX53VG 137642650 Ki = 38 nM T68706 CHI60U 137642806 Ki = 0.7 nM T68706 C7W9US 137643496 Ki = 1.1 nM T68706 C7PR9K 137644391 Ki = 1.5 nM T68706 C98VOE 137645351 Ki = 1.5 nM T68706 C0NWD3 137645581 Ki = 15 nM T68706 CQ6SI9 137645677 Ki = 7 nM T68706 CJT5C4 137646929 Ki = 4 nM T68706 C8WED4 137647032 Ki = 0.9 nM T68706 C76BDY 137647768 Ki = 8 nM T68706 CD3CZ6 137647834 Ki = 3 nM T68706 C64QUK 137648887 Ki = 50 nM T68706 CBP37G 137649385 Ki = 7 nM T68706 C2N9LT 137650514 Ki = 6 nM T68706 COR8J3 137652054 Ki = 27 nM T68706 CJX57S 137652059 Ki = 4 nM T68706 CVC56D 137652453 Ki = 11 nM T68706 CUP70F 137652558 Ki = 3.4 nM T68706 CJVG81 137652912 Ki = 23 nM T68706 CPO80U 137653066 Ki = 5 nM T68706 CN5VC7 137653379 Ki = 8.1 nM T68706 C34XTZ 137653755 Ki = 2 nM T68706 CUHM58 137653788 Ki = 3 nM T68706 C4B8DK 137654788 Ki = 9 nM T68706 C4XTJ7 137655341 Ki = 1.4 nM T68706 C7W1GU 137655527 Ki = 4 nM T68706 CBRA14 137655621 Ki = 4.7 nM T68706 CI78BN 137656445 Ki = 3 nM T68706 CD9N0S 137656589 Ki = 8 nM T68706 CV7T5U 137656624 Ki = 16.7 nM T68706 CI3A4J 137657514 Ki = 1.1 nM T68706 CO09SX 137658594 Ki = 3 nM T68706 CZY51S 137659359 Ki = 0.6 nM T68706 C8J2FS 137659865 Ki = 1 nM T68706 CXYA13 137660373 Ki = 2.4 nM T68706 C37WVK 137660935 Ki = 18 nM T68706 CGBP12 137661234 Ki = 3.1 nM T68706 CSI79D 137661408 Ki = 4 nM T68706 CV3NU9 137661582 Ki = 4.8 nM T68706 CDP9F6 145979561 Ki = 41 nM T68706 C0FVL7 145980400 Ki = 825 nM T68706 C7U6AC 145980921 Ki = 60 nM T68706 C1PY3D 145982564 Ki = 2600 nM T68706 C0F2HS 145982570 Ki = 290 nM T68706 C9BAM3 145982642 Ki = 2500 nM T68706 CO1L7J 145982755 Ki = 260 nM T68706 CH49CQ 145982874 Ki = 700 nM T68706 CL4F2V 145983062 Ki = 74 nM T68706 C8P4IY 145983083 Ki = 280 nM T68706 CD4V6Y 145983456 Ki = 100 nM T68706 C0VPE7 145983531 Ki = 990 nM T68706 CMN3C0 145983800 Ki = 210 nM T68706 CKY29N 145984016 Ki = 140 nM T68706 C71KAW 145984052 Ki = 140 nM T68706 C7Y5TR 145984180 Ki = 330 nM T68706 CI2E5Y 145984243 Ki = 74 nM T68706 CP4M8O 145984298 Ki = 130 nM T68706 CR0E5D 145984449 Ki = 130 nM T68706 CBK18Y 145984711 Ki = 110 nM T68706 C9W1TO 145984728 Ki = 80 nM T68706 CZ9MK3 145984956 Ki = 990 nM T68706 C6VYO5 145985131 Ki = 500 nM T68706 C0DJ8X 145985285 Ki = 170 nM T68706 CME81P 145985674 Ki = 3000 nM T68706 CMT30D 145985833 Ki = 64 nM T68706 CN96XK 145985989 Ki = 200 nM T68706 C6UA9H 145986239 Ki = 190 nM T68706 CG7LW4 145987687 Ki = 38 nM T68706 C3C2LW 145989654 Ki = 614 nM T68706 C4IW1B 145989737 Ki = 240 nM T68706 C4ACG5 145990382 Ki = 600 nM T68706 CZJY41 145990864 Ki = 21.5 nM T68706 CB9FH7 145992096 Ki = 250 nM T68706 C9KC4Q 145993075 Ki = 60 nM T68706 D05JJL 44584947 Ki = 23 nM T68706 D0A6FZ 75593419 Ki = 4.3 nM T68706 D0Y9PH 45486355 Ki = 0.81 nM T67977 D00UVA 11556711 IC50 = 490 nM T67977 D06OMK 445643 Ki = 360 nM T67977 D09HNR 3002190 Ki = 2.4 nM T67977 D0N3VR 71616 Ki = 660 nM T67977 D0A7ZK 56944144 IC50 > 20000 nM T67977 D0G7UX 5284373 Ki = 980 nM T67977 CC92YE 11755033 IC50 > 100000 nM T67977 CB8E2S 45482734 Ki = 1.2 nM T67977 CDM1L4 45482735 Ki = 5.6 nM T67977 CEM05T 45482739 Ki = 5.3 nM T67977 C2LU1K 45482740 Ki = 25 nM T67977 CS9OV5 71315139 IC50 = 330 nM T67977 CDJ93N 118753464 IC50 = 1800 nM T67977 CC43OQ 134149366 IC50 > 50000 nM T67977 C7GP2R 136123532 Ki = 24 nM T67977 C8V9ER 137440575 IC50 = 25900 nM T67977 CZE16B 146026197 IC50 = 36600 nM T67977 C28HEF 155519544 IC50 > 62200 nM T49989 D06TFI 10090485 IC50 = 1300 nM T49989 D0Z1DH 10029385 IC50 > 1200 nM T49989 C47NLO 2869892 IC50 = 830 nM T49989 C31FHN 5330788 IC50 > 20000 nM T49989 CK2Q0Y 9972086 IC50 = 8730 nM T49989 CZV48E 9972935 IC50 > 20000 nM T49989 CU3D9T 9973794 IC50 > 20000 nM T49989 C6UJ3H 9995838 IC50 = 19630 nM T49989 CPZ34K 10002593 IC50 > 20000 nM T49989 C1XVD4 10049774 IC50 = 14540 nM T49989 C69VRQ 10064294 IC50 = 395 nM T49989 C1TXC3 10094943 IC50 > 20000 nM T49989 CQP2T6 10321041 IC50 > 20000 nM T49989 CZV97C 10359218 IC50 = 668 nM T49989 C8X2RY 10456042 IC50 = 19750 nM T49989 C30PKR 11248978 IC50 = 2000 nM T49989 CSXY78 11294864 IC50 = 3100 nM T49989 CPU9I3 11316975 IC50 > 20000 nM T49989 CQ8I4H 11328863 IC50 > 20000 nM T49989 CC96QB 11507696 IC50 > 20000 nM T49989 CYQ4O9 11723225 IC50 = 1300 nM T49989 CE9MU4 11740079 IC50 = 690 nM T49989 CPQ31L 25195294 IC50 = 140.4 nM T49989 CN2QG1 44223357 IC50 = 236 nM T49989 CSBC59 44396134 IC50 = 9500 nM T49989 CB5NF6 44408672 IC50 > 20000 nM T49989 CYG2F3 44408807 IC50 > 20000 nM T49989 CM54AI 44408849 IC50 > 20000 nM T49989 CN4X1A 44408884 IC50 = 10840 nM T49989 C2Q0GE 50990922 IC50 = 2000 nM T49989 C91FTP 57339386 IC50 = 16 nM T49989 CIP7B1 60182373 IC50 = 38 nM T49989 CQ6KV9 60182388 IC50 = 327 nM T49989 CV63UL 67240318 IC50 > 10000 nM T49989 CC9V0P 121411739 IC50 > 15000 nM T49989 C9CV7H 121411850 IC50 = 7600 nM T49989 CT9NY8 121411862 IC50 = 730 nM T49989 C09YCI 121411874 IC50 = 40 nM T49989 C9HV3A 121411904 IC50 > 15000 nM T49989 CC4SD7 121411952 IC50 = 7 nM T49989 C2U3DY 121411994 IC50 = 14000 nM T49989 CC2H7S 121412004 IC50 = 14000 nM T49989 C7JS3L 121412028 IC50 > 15000 nM T49989 CU3BI0 121412063 IC50 = 4300 nM T49989 CLW35N 121412124 IC50 = 390 nM T49989 CIHA53 122510417 IC50 > 15000 nM T49989 COX7E3 122510453 IC50 > 15000 nM T49989 C26UNE 122510498 IC50 > 15000 nM T49989 CM6Q5H 122510766 IC50 = 5710 nM T49989 C0TZE4 122510927 IC50 = 2930 nM T49989 CYE69W 126484202 IC50 = 810 nM T49989 CUO92C 126484344 IC50 > 15000 nM T49989 C8D2RG 126499376 IC50 = 550 nM T49989 C9MUH4 126499699 IC50 = 8500 nM T49989 CP7DF4 126499823 IC50 = 110 nM T49989 C5K8PR 126499902 IC50 > 15000 nM T49989 CWD1V7 126499983 IC50 > 15000 nM T49989 CPK6O7 126537450 IC50 > 15000 nM T49989 CM42SX 126537451 IC50 = 940 nM T49989 CYQ24M 126537506 IC50 = 310 nM T49989 C3WGZ0 126622458 IC50 = 1100 nM T49989 C5H8LU 126677289 IC50 = 1100 nM T49989 CJPO36 135223028 IC50 = 820 nM T49989 C5QF0M 135233366 IC50 = 12900 nM T49989 C4N6OZ 135262129 IC50 > 15000 nM T49989 CZAN82 135262182 IC50 = 77 nM T49989 CQ9B5Y 135262208 IC50 = 2000 nM T49989 C6YJF9 135262382 IC50 = 3000 nM T49989 CV72CD 135262410 IC50 = 570 nM T49989 CPT0V7 138454752 IC50 = 698 nM T49989 C2MD1Q 155513187 IC50 > 10000 nM T49989 D05NEC 60182364 IC50 = 15 nM T49989 D06BDC 10361101 IC50 = 352 nM T49989 D06KKN 11655119 IC50 = 190 nM T49989 D0C7WP 4521392 IC50 = 66 nM T49989 D0F2MP 60182389 IC50 = 26 nM T49989 D0PP6Y 60182393 IC50 = 1.37 nM T49989 D0XB4P 447966 IC50 = 400 nM T49989 D0Y0BK 11524144 IC50 = 102.9 nM T28887 D00SQN 12136798 IC50 = 833 nM T28887 D07POC 176870 IC50 > 32000 nM T28887 D08CDI 208908 IC50 > 10000 nM T28887 D0E3SH 6918837 IC50 = 19.79 nM T28887 D0E7PQ 5311 IC50 = 5.5 nM T28887 D0L7LC 5352062 Ki = 0.15 nM T28887 D0Y3KG 3121 IC50 = 103000 nM T28887 D00FHR 9865515 IC50 = 35000 nM T28887 D05KED 53340666 IC50 = 100 nM T28887 D07FPY 6918877 Ki = 82 nM T28887 D09XIZ 11538455 Ki = 0.5 nM T28887 D0B3FV 6445533 Ki = 340 nM T28887 D0B7CH 4775 IC50 = 93000 nM T28887 D0E6UZ 54575456 IC50 = 1.4 nM T28887 D0GE5B 56654642 IC50 = 10700 nM T28887 D0GH3Q 9804992 Ki = 39 nM T28887 D0L2UQ 49855250 Ki = 16 nM T28887 D0M8FD 4261 IC50 = 9884 nM T28887 D0V0SL 11749858 Ki = 280 nM T28887 D0XT6W 6918638 Ki = 22 nM T28887 D0Z4RC 24756910 IC50 = 79.8 nM T28887 D0J8OC 5186 Ki = 105 nM T28887 D00HXJ 118884610 Ki = 173 nM T28887 D0CH8Q 56965342 IC50 > 10000 nM T28887 D0L1NO 72722126 IC50 = 280 nM T28887 D0N2DK 72710871 IC50 = 32.9 nM T28887 D0QX3G 71532921 IC50 = 2800 nM T28887 D0YN2T 86302836 IC50 = 6700 nM T28887 D0ZG5X 71811260 IC50 = 99 nM T28887 D0N3SH 4996 Ki = 1000 nM T28887 D0W9NH 2746 IC50 > 20000 nM T28887 CCK23B 4144 IC50 = 100 nM T28887 CBIR94 10313 IC50 = 1920 nM T28887 CL25FN 76175 IC50 > 30000 nM T28887 C1N2KZ 88129 IC50 = 39000 nM T28887 CE69VZ 148031 IC50 = 582.3 nM T28887 CW70DI 211808 IC50 > 100000 nM T28887 CF60JA 220184 IC50 = 11620 nM T28887 CH1JD3 419176 IC50 = 26000 nM T28887 C0Y4WC 614947 Ki = 811.5 nM T28887 C0EM9B 801008 IC50 = 3100 nM T28887 CU3HS2 1108280 IC50 > 100000 nM T28887 CA9TW1 2723947 IC50 = 3675 nM T28887 CK8I3T 3432579 IC50 = 3720 nM T28887 CZA83Y 4118131 IC50 = 2350 nM T28887 CV9JS5 4288771 IC50 = 3300 nM T28887 C9OQP1 4548286 IC50 = 70.2 nM T28887 CH5FO1 5353767 IC50 = 200 nM T28887 CXUP49 5353769 IC50 = 600 nM T28887 C1RD7E 6918878 IC50 > 10000 nM T28887 CE9LP2 9543539 IC50 = 5000 nM T28887 CJ07ZA 9800555 IC50 > 32000 nM T28887 CC0EU7 9828788 IC50 = 25 nM T28887 CH2LR4 9835152 IC50 = 1030 nM T28887 CLYJ85 9848223 IC50 = 800 nM T28887 C4GBE9 9860473 IC50 = 63 nM T28887 CSW4Y1 9891541 IC50 = 690 nM T28887 C81EYJ 9923508 IC50 = 1619.7 nM T28887 CQG4V8 9924543 IC50 = 779 nM T28887 COLN58 9965621 IC50 = 1150 nM T28887 CTYI59 9977701 IC50 = 2800 nM T28887 CDT7U0 9998313 IC50 = 50 nM T28887 CR98AV 9999602 IC50 = 310 nM T28887 C0S5TP 10012466 IC50 = 500 nM T28887 CXA5J1 10068980 IC50 = 120 nM T28887 CCD3S6 10090483 IC50 = 40 nM T28887 CX81ML 10092736 IC50 = 4600 nM T28887 CWA9R2 10135838 IC50 > 32000 nM T28887 CL4C9H 10154438 Ki = 0.1 nM T28887 CB2OV7 10266393 IC50 = 100 nM T28887 C7RC1E 10309899 IC50 = 27 nM T28887 C5S8XH 10340474 IC50 = 400 nM T28887 C1G9YS 10362929 IC50 = 50 nM T28887 CN5IT3 10381402 IC50 = 40 nM T28887 C9OU5F 10464879 Ki = 12.81 nM T28887 CW2X8Z 10474722 IC50 = 2200 nM T28887 CX60YL 10502119 IC50 > 100000 nM T28887 CX2KA5 10572471 IC50 > 100000 nM T28887 CDY91S 10584105 Ki = 0.53 nM T28887 CAYN96 10597715 IC50 = 40000 nM T28887 C3N9BM 10643236 IC50 > 100000 nM T28887 C9VCT3 10669053 IC50 = 44000 nM T28887 CSMT47 10728039 Ki = 83.8 nM T28887 CQZ36O 10785752 IC50 > 100000 nM T28887 CD0G3L 10832425 IC50 > 100000 nM T28887 CKS03P 10834447 IC50 = 6000 nM T28887 C80ZXG 10881097 IC50 = 35 nM T28887 CAF1N8 10906013 IC50 = 504700 nM T28887 CK8UV7 11019840 Ki = 1.47 nM T28887 CX50LC 11066195 IC50 = 103 nM T28887 CW2GJ0 11166750 IC50 = 63 nM T28887 CFEN82 11177718 IC50 = 50 nM T28887 C5JR3Q 11184660 IC50 > 10000 nM T28887 CMQ38G 11199235 IC50 = 100 nM T28887 CA48NR 11199635 IC50 = 41 nM T28887 C8G5WP 11210533 IC50 = 2100 nM T28887 CG27ZR 11212396 IC50 = 25 nM T28887 C89SVA 11223999 IC50 = 20 nM T28887 CYJ60V 11244651 IC50 = 119700 nM T28887 CSO06H 11259022 IC50 = 79 nM T28887 CI7W3O 11267278 IC50 = 10200 nM T28887 C6AKW1 11270791 IC50 = 50 nM T28887 CM6ZW2 11279156 IC50 = 19100 nM T28887 CV9Y4T 11326181 IC50 = 200 nM T28887 C0L1BK 11357542 IC50 > 40000 nM T28887 CZT79Q 11360420 IC50 = 31 nM T28887 C0V2DZ 11370695 IC50 > 40000 nM T28887 CY34EQ 11393847 IC50 > 20000 nM T28887 C9QB0C 11396478 IC50 = 16 nM T28887 CVH8N1 11430412 IC50 = 79 nM T28887 CRTV86 11430535 IC50 = 63 nM T28887 CNU8D3 11438971 IC50 = 100 nM T28887 C5HP1B 11441977 IC50 = 20 nM T28887 CMB9R2 11452638 IC50 = 328 nM T28887 C3BGS1 11473639 IC50 = 75 nM T28887 CB3N5M 11514394 IC50 = 689 nM T28887 CRZ7H2 11556677 IC50 > 10000 nM T28887 C2F9NT 11558827 IC50 = 1740 nM T28887 C9UN7F 11637884 IC50 = 50 nM T28887 C24SBP 11657529 IC50 > 5000 nM T28887 CQ32FV 11664499 IC50 = 200 nM T28887 CG9OC4 11682502 IC50 = 30 nM T28887 CYB26W 11688197 IC50 = 245 nM T28887 C8N9UZ 11724319 IC50 = 300 nM T28887 C9Y2GM 11794739 IC50 > 100000 nM T28887 C58FZA 11795873 IC50 = 7700 nM T28887 CE4Z0Y 11844891 IC50 = 44000 nM T28887 C9G1BN 11993595 IC50 = 730 nM T28887 CH5JS7 11993694 IC50 = 180 nM T28887 C1BVY9 12325934 IC50 > 30000 nM T28887 CR5F6I 12397856 IC50 = 9500 nM T28887 CJ94OC 12542182 Ki = 7.87 nM T28887 C06UTF 13507024 IC50 = 790 nM T28887 CVH7N1 13746652 IC50 = 110500 nM T28887 C4XJ8M 13889849 Ki = 10500 nM T28887 C1KR4L 14113324 IC50 = 21000 nM T28887 C15MQN 14113325 IC50 = 3200 nM T28887 C2D1KP 15983982 Ki = 136 nM T28887 CHB82E 15986417 IC50 = 6960 nM T28887 C52EVH 15986418 IC50 = 162 nM T28887 CS1QO9 15986509 IC50 = 69.8 nM T28887 C5T1WF 16006672 IC50 > 10000 nM T28887 CQGC05 16036765 IC50 = 3000 nM T28887 CM3T2E 16049824 IC50 > 1 nM T28887 C30UFT 16066811 IC50 = 16720 nM T28887 CFK8J5 16068056 Ki = 65 nM T28887 CMQP70 16068495 Ki = 78 nM T28887 CT84XO 16068594 Ki = 57 nM T28887 CF3ZG5 16068595 Ki = 54 nM T28887 CL60CA 16068912 Ki = 94 nM T28887 C9ZQB3 16095102 Ki > 5000 nM T28887 C6RE2F 16220721 Ki = 5.32 nM T28887 C6BGM2 16659535 IC50 = 420 nM T28887 CQI9N3 16659537 IC50 = 730 nM T28887 C5YFV9 16661453 IC50 = 1190 nM T28887 C8S5OX 16661455 IC50 = 520 nM T28887 CH67WF 16661458 IC50 = 210 nM T28887 CZ72YC 16661613 IC50 = 530 nM T28887 C8DZ1T 16661615 IC50 = 1150 nM T28887 CQV40I 16661617 IC50 = 250 nM T28887 C5CIB4 16663079 IC50 > 50000 nM T28887 CUG50I 16733294 IC50 = 1600 nM T28887 CWO7V0 16733295 IC50 = 3410 nM T28887 C4W0PG 16733410 IC50 = 1720 nM T28887 C0MO3Z 16733411 IC50 = 4090 nM T28887 C3QL4X 16733412 IC50 > 30000 nM T28887 CV54SY 16733414 IC50 = 6120 nM T28887 C1VCX2 16733415 IC50 = 1050 nM T28887 CXN07K 16733416 IC50 = 13900 nM T28887 CP9AR8 16733417 IC50 = 2060 nM T28887 CUE62T 16733590 IC50 = 12300 nM T28887 CF7JR0 17756401 IC50 = 32 nM T28887 C3FN8M 17756403 IC50 = 79 nM T28887 C5P8QU 18618646 IC50 = 1000 nM T28887 C9FL1J 18618663 IC50 = 1000 nM T28887 CQHD27 20459443 IC50 = 431 nM T28887 C2X5PQ 22958841 IC50 = 940 nM T28887 CD2L0V 22986769 IC50 = 300 nM T28887 C1EG3M 22986772 IC50 = 100 nM T28887 CSM54L 22986780 IC50 = 100 nM T28887 CE3T2V 22986786 IC50 = 600 nM T28887 C2HZ8N 22986792 IC50 = 840 nM T28887 CO8B1H 22986803 IC50 = 2400 nM T28887 CN64IA 22986815 IC50 = 2000 nM T28887 CD16PI 23521584 IC50 = 1900 nM T28887 CEF8W4 23625604 IC50 = 15848.93 nM T28887 CB8A5Q 23648260 IC50 = 31738 nM T28887 C36NKL 23648268 IC50 > 20000 nM T28887 C5YBX0 23760408 IC50 = 110 nM T28887 CM73VT 23818230 IC50 = 290 nM T28887 CVAB64 23846833 IC50 = 23 nM T28887 C8RC9P 24744325 IC50 = 20000 nM T28887 C17GDO 24779722 IC50 = 331 nM T28887 CIO7Q6 24853792 IC50 > 10000 nM T28887 CBN0J5 24853793 IC50 > 1 nM T28887 CLT5J2 24881257 IC50 = 3970 nM T28887 C5GCM1 24881328 IC50 = 797 nM T28887 C8QVB1 24881329 IC50 = 3130 nM T28887 CU0AM3 24881330 IC50 = 1990 nM T28887 CQM51L 24881331 IC50 = 2780 nM T28887 C4KH8F 24881332 IC50 = 2010 nM T28887 C1KA3V 24881333 IC50 = 737 nM T28887 C47APB 24881402 IC50 = 433 nM T28887 CSN8W1 24881403 IC50 = 942 nM T28887 C1UQ3K 24881404 IC50 = 1970 nM T28887 C51TMH 24881405 IC50 = 552 nM T28887 C9EZI7 24881406 IC50 = 440 nM T28887 C6P3HS 24881407 IC50 = 790 nM T28887 CZ3TU1 24881464 IC50 = 518 nM T28887 CDI49N 24881465 IC50 = 529 nM T28887 CQGP87 24881466 IC50 = 406 nM T28887 CS1MH8 24888322 IC50 = 22000 nM T28887 CC0R9O 24938735 IC50 = 3.8 nM T28887 CF03HD 24948905 IC50 = 3650 nM T28887 CHP8O6 24948906 IC50 = 938 nM T28887 C1KRT8 24948907 IC50 = 3430 nM T28887 CKY2P8 24948908 IC50 = 3458 nM T28887 C25CFI 24948909 IC50 = 2830 nM T28887 CWQ04Z 24948910 IC50 = 4900 nM T28887 CM9I3X 24951310 IC50 = 3320 nM T28887 CX1YF8 24951311 IC50 = 3580 nM T28887 CV10XU 24951312 IC50 = 8104 nM T28887 CD6KV0 24951313 IC50 = 5810 nM T28887 CQY9Z0 24951314 IC50 = 6851 nM T28887 CV8EF6 25032862 IC50 > 50000 nM T28887 CX69SY 25066355 IC50 = 643 nM T28887 CF8VP4 25066356 IC50 = 1100 nM T28887 CS9XH7 25066547 IC50 = 286 nM T28887 C46AGN 25066548 IC50 = 119 nM T28887 CJF2M7 25066549 IC50 = 444 nM T28887 CY9JV6 25113671 IC50 = 1390 nM T28887 CH7TV1 25150907 IC50 = 4750 nM T28887 CH1LV3 25150908 IC50 = 4420 nM T28887 C4GC5R 25151496 IC50 = 994 nM T28887 CFO6B0 25151497 IC50 = 1020 nM T28887 COGD60 25151676 IC50 = 6780 nM T28887 CTP21Q 25151864 IC50 = 1890 nM T28887 CWL8E0 25151865 IC50 = 10550 nM T28887 CWR7N3 25152061 IC50 = 5880 nM T28887 C4C6AM 25152063 IC50 = 3740 nM T28887 C4I1CJ 25155417 IC50 > 20000 nM T28887 CB4E2J 25155956 IC50 > 50000 nM T28887 C74IYD 25190760 IC50 = 3990 nM T28887 CO14XG 25195084 IC50 > 10000 nM T28887 CE5F2V 25195975 IC50 = 710 nM T28887 CCD5M7 25227504 IC50 = 198 nM T28887 CK0D5S 25227505 IC50 = 206 nM T28887 CN97JP 25227508 IC50 = 136 nM T28887 CW8R1B 25227513 IC50 = 90.7 nM T28887 CE0NV4 25257993 IC50 = 341.3 nM T28887 C43BHY 25269097 IC50 = 9300 nM T28887 CN7K1S 25374100 IC50 = 620 nM T28887 CU53WB 42596953 IC50 = 630 nM T28887 CJ1RQ7 42598706 IC50 = 376 nM T28887 C2LES7 42599455 IC50 = 2116.3 nM T28887 C2KO0F 42599456 IC50 = 2028.3 nM T28887 C1UAO7 42601485 IC50 = 37000 nM T28887 COI7Y3 42611300 IC50 = 2200 nM T28887 CU23PG 42611301 IC50 = 130 nM T28887 C3ZV9H 42611302 IC50 = 2700 nM T28887 CW1G2R 42611390 IC50 = 15 nM T28887 C62QFJ 42611486 IC50 = 2000 nM T28887 CQ37HN 42612743 IC50 = 255.3 nM T28887 CLH2Q7 42612852 IC50 = 2300 nM T28887 CQB20M 42630929 IC50 = 1700 nM T28887 CDT65Y 42631047 IC50 = 1560 nM T28887 C2NF6U 42632370 IC50 = 320 nM T28887 C9B8VR 42632614 IC50 > 5000 nM T28887 CB79DG 42637299 IC50 > 100000 nM T28887 CP36KB 42637300 IC50 > 100000 nM T28887 CI8J6H 42637372 IC50 = 6600 nM T28887 C5RYO0 42637373 IC50 > 100000 nM T28887 CJ0CG5 42638004 IC50 > 100000 nM T28887 C8X0TG 42638005 IC50 = 23000 nM T28887 C3LHF9 42917485 IC50 = 970 nM T28887 CO57GS 44138033 IC50 = 603 nM T28887 C7RCY4 44178890 IC50 = 110 nM T28887 CY0QB9 44253226 IC50 = 1760 nM T28887 CL80GX 44328682 IC50 = 900 nM T28887 C86IOC 44328927 IC50 > 10000 nM T28887 C7G5CO 44359547 IC50 = 780 nM T28887 CIT7A9 44359548 IC50 = 9700 nM T28887 CUM0Q6 44359555 IC50 = 650 nM T28887 CP92JV 44359673 IC50 > 100000 nM T28887 CQ7J2G 44359674 IC50 = 2800 nM T28887 CGK71T 44359675 IC50 = 4000 nM T28887 C2V4DN 44359681 IC50 = 7000 nM T28887 CX31TB 44359788 IC50 = 6800 nM T28887 CQ5Y8G 44359800 IC50 > 100000 nM T28887 CL82CH 44359814 IC50 > 100000 nM T28887 C5YRC9 44431499 IC50 = 1200 nM T28887 CNC51G 44447194 IC50 > 50000 nM T28887 C5VP4D 44454144 IC50 > 50000 nM T28887 C8A1ZD 44456564 IC50 = 140 nM T28887 CT19ZV 44456601 IC50 = 38 nM T28887 CJ0L4C 44456965 IC50 = 3000 nM T28887 C58YCH 44456972 IC50 > 40000 nM T28887 CY4I7R 44456994 IC50 > 40000 nM T28887 C5HS2K 44456995 IC50 > 10000 nM T28887 CPDE25 44507029 IC50 = 29 nM T28887 CBL69N 44507542 IC50 = 52 nM T28887 C7F8YJ 44543715 Ki = 600 nM T28887 CIL9F4 44549342 IC50 = 37400 nM T28887 CQ2TU3 44550557 Ki = 6590 nM T28887 CEM91G 44562802 IC50 = 220 nM T28887 CG9OD1 44571302 IC50 = 640 nM T28887 C0ZX1A 44571330 IC50 = 2340 nM T28887 CY83MO 44571331 IC50 = 1210 nM T28887 CP6D1G 44571332 IC50 = 440 nM T28887 COM65J 44572384 IC50 >= 25000 nM T28887 CA6Q9Y 44592060 IC50 = 127 nM T28887 CE5W3U 44598288 IC50 = 530 nM T28887 C68BJH 44598289 IC50 = 2670 nM T28887 C9K2WV 44598290 IC50 = 870 nM T28887 C16ZEP 44598291 IC50 = 150 nM T28887 C28GHB 44598344 IC50 = 1400 nM T28887 CU65LR 44598345 IC50 = 607 nM T28887 CHQ86X 44598347 IC50 = 1400 nM T28887 CCVA51 44598385 IC50 = 1380 nM T28887 C29NXL 44598386 IC50 = 6700 nM T28887 CK8V9I 44598388 IC50 = 240 nM T28887 C3TOK2 44598431 IC50 = 1000 nM T28887 CPZ65Q 44598479 IC50 = 7040 nM T28887 CGT51H 44598480 IC50 = 4900 nM T28887 CZ62IW 44598481 IC50 > 10000 nM T28887 C0OT6I 44598482 IC50 = 6050 nM T28887 CX8U6S 44598483 IC50 = 9700 nM T28887 C5H8RA 44598536 IC50 > 10000 nM T28887 CC2QV9 44623002 IC50 = 1500 nM T28887 CVJ51M 44623152 IC50 = 1000 nM T28887 C6TJ2G 44623153 IC50 = 1300 nM T28887 C42SJP 45141750 IC50 = 523 nM T28887 CLE9U5 45141751 IC50 = 336 nM T28887 C09NQK 45269071 IC50 = 52560 nM T28887 CIWD29 45269932 IC50 = 11250 nM T28887 CY25MX 45270754 IC50 = 12250 nM T28887 CSM1O6 45271073 IC50 = 74000 nM T28887 CP2XO6 45272484 IC50 = 9650 nM T28887 CL71OI 45483433 IC50 = 3503 nM T28887 CUF94Q 45483434 IC50 = 1528 nM T28887 C4S2PN 45483435 IC50 = 1243 nM T28887 C9RIM5 45484125 Ki = 2430 nM T28887 C7EAV5 45485820 IC50 = 150 nM T28887 C2M4GV 46179732 IC50 = 1190 nM T28887 CS75CD 46179779 IC50 = 4180 nM T28887 C39YKM 46179780 IC50 = 2750 nM T28887 C0CKE5 46180624 IC50 > 30000 nM T28887 C7GYH0 46180758 IC50 = 12000 nM T28887 C27IKH 46180759 IC50 > 30000 nM T28887 CSC1Y9 46180760 IC50 = 5220 nM T28887 C70FSJ 46180763 IC50 = 1320 nM T28887 C0W8DB 46187719 IC50 = 950 nM T28887 CV7D4Z 46187885 IC50 = 830 nM T28887 C53ZSX 46187886 IC50 = 3170 nM T28887 CEV52J 46187887 IC50 = 710 nM T28887 CSC70G 46187888 IC50 = 2080 nM T28887 C7SC8A 46187889 IC50 = 1030 nM T28887 CQLG06 46187890 IC50 = 1860 nM T28887 CVGN05 46187891 IC50 = 3190 nM T28887 CF29IN 46188075 IC50 = 760 nM T28887 COWJ59 46190552 IC50 = 200 nM T28887 C8YO4W 46190553 IC50 = 1250 nM T28887 CEX48K 46190554 IC50 = 860 nM T28887 C6J9DI 46190555 IC50 = 230 nM T28887 C53RNX 46190556 IC50 = 8260 nM T28887 CPS37G 46190557 IC50 = 350 nM T28887 C2MOT0 46190609 IC50 = 380 nM T28887 CJ8OT2 46190610 IC50 = 1360 nM T28887 CX93ZQ 46190753 IC50 = 2050 nM T28887 C85WSJ 46190754 IC50 > 10000 nM T28887 C9VEX6 46190755 IC50 > 10000 nM T28887 C6O5AD 46190756 IC50 = 2560 nM T28887 C7F8AM 46190820 IC50 > 10000 nM T28887 C8JY0S 46190821 IC50 = 3650 nM T28887 CUCK61 46190822 IC50 = 2380 nM T28887 CXQ51Y 46190823 IC50 = 5390 nM T28887 CR0G9O 46190824 IC50 = 1830 nM T28887 CDP80X 46190825 IC50 = 1920 nM T28887 C3ETP2 46190826 IC50 = 8760 nM T28887 CD57RJ 46197798 IC50 = 217 nM T28887 CR04HA 46197799 IC50 = 364 nM T28887 C3ZE2B 46198177 IC50 = 1272 nM T28887 CQ83FI 46203315 IC50 > 10000 nM T28887 CK8YL5 46203316 IC50 = 8390 nM T28887 C1YB9P 46203618 IC50 > 10000 nM T28887 C4I5DH 46203619 IC50 > 10000 nM T28887 C43KVC 46203620 IC50 > 10000 nM T28887 CY7ER9 46203621 IC50 > 10000 nM T28887 CW13ZY 46203622 IC50 > 10000 nM T28887 CND31M 46203623 IC50 > 10000 nM T28887 C1RX2K 46203949 IC50 > 10000 nM T28887 CZJ86R 46203950 IC50 > 10000 nM T28887 CNA07J 46203951 IC50 > 10000 nM T28887 CQ69AM 46205433 IC50 = 113 nM T28887 C74YBE 46228450 IC50 = 1650 nM T28887 CT12IM 46228452 IC50 = 3820 nM T28887 CP0M5Z 46228453 IC50 = 4000 nM T28887 C70TRH 46228455 IC50 = 4130 nM T28887 C5ZLO9 46228500 IC50 = 1770 nM T28887 CZ2AN4 46228502 IC50 = 3620 nM T28887 C2V0HA 46228503 IC50 = 2560 nM T28887 CY5M3P 46228505 IC50 = 3230 nM T28887 CS2T4I 46228518 IC50 = 1170 nM T28887 CHD8I4 46228520 IC50 = 3200 nM T28887 C83OSG 46228521 IC50 = 3780 nM T28887 C9W8DC 46228523 IC50 = 3390 nM T28887 CBU85J 46228543 IC50 = 1550 nM T28887 CB23XN 46228545 IC50 = 3340 nM T28887 CN5ES6 46228546 IC50 = 4250 nM T28887 CRQ2O6 46228548 IC50 = 1060 nM T28887 C4P0JQ 46228579 IC50 = 1980 nM T28887 CU5K1N 46228581 IC50 = 2210 nM T28887 CDRB91 46228582 IC50 = 3020 nM T28887 C28HRA 46228584 IC50 = 3540 nM T28887 CYR6A2 46228609 IC50 = 4420 nM T28887 CB3AD0 46228611 IC50 = 5770 nM T28887 CBW7X1 46228612 IC50 = 4580 nM T28887 CVO6R0 46228614 IC50 = 12170 nM T28887 COP28Q 46228637 IC50 = 580 nM T28887 CUKY04 46228882 IC50 = 1290 nM T28887 CDV6P0 46228884 IC50 = 8210 nM T28887 CEAT10 46228885 IC50 = 3410 nM T28887 C5FT7A 46228887 IC50 = 5100 nM T28887 C9VTZ7 46228937 IC50 = 2670 nM T28887 COH42M 46228939 IC50 = 4070 nM T28887 C4FWS2 46228940 IC50 = 1000 nM T28887 CWS34O 46228942 IC50 = 5570 nM T28887 CN8F9S 46830326 IC50 = 160 nM T28887 CKIP01 46846372 IC50 = 197 nM T28887 C4NLH6 46846374 IC50 = 120 nM T28887 C8D4XL 46861823 IC50 = 27600 nM T28887 CQTI31 46881225 IC50 > 30000 nM T28887 CM9W8B 46886948 IC50 = 63 nM T28887 C3X1PB 46886949 IC50 = 25 nM T28887 CA8ZB0 46886950 IC50 = 25 nM T28887 C5STW2 46887022 IC50 = 20 nM T28887 C35ATX 46887023 IC50 = 16 nM T28887 C35LCR 46887024 IC50 = 160 nM T28887 C1C7TX 46887025 IC50 = 120 nM T28887 CC6I4F 46887026 IC50 = 120 nM T28887 CEMV64 46887060 IC50 = 200 nM T28887 CCU65S 46887061 IC50 = 160 nM T28887 C24FTM 46887062 IC50 = 120 nM T28887 C8VD6Z 46887093 IC50 = 160 nM T28887 C3UNV6 46887094 IC50 = 50 nM T28887 CJE6Q2 46887127 IC50 = 31 nM T28887 C4OWH7 46887128 IC50 = 31 nM T28887 C74SPT 46887178 IC50 = 100 nM T28887 C9I6NF 46887179 IC50 = 50 nM T28887 C28RSA 46887180 IC50 = 40 nM T28887 CH85NX 46887211 IC50 = 79 nM T28887 C8YAV5 46887212 IC50 = 50 nM T28887 CJ30VB 46887241 IC50 = 100 nM T28887 CX53HE 46887282 IC50 = 500 nM T28887 CU38FK 46887283 IC50 = 400 nM T28887 C0CTM9 46887332 IC50 = 100 nM T28887 CP4W7O 46887556 IC50 = 50 nM T28887 C2GP9T 46887557 IC50 = 160 nM T28887 C3UIY6 46887558 IC50 = 63 nM T28887 CUR2X5 46887559 IC50 = 200 nM T28887 CMU9D7 46887584 IC50 = 100 nM T28887 CA8JT1 46887585 IC50 = 63 nM T28887 C93CLK 46887919 IC50 = 23000 nM T28887 CPSI47 46890583 Ki = 315 nM T28887 C90NYX 46896338 IC50 > 30000 nM T28887 C1HV6U 46907409 IC50 > 20000 nM T28887 CY7B1U 46913905 IC50 = 620 nM T28887 C42UBP 46913906 IC50 = 825 nM T28887 CWA0M8 46916092 IC50 = 796.2 nM T28887 CYN9W5 46916093 IC50 = 210 nM T28887 C78XOJ 46916094 IC50 = 580 nM T28887 CXH64A 46918825 IC50 = 3981.07 nM T28887 C1F4VZ 49798604 IC50 = 43160 nM T28887 CL7PS1 49831258 IC50 = 2100 nM T28887 CI5L2P 49846123 IC50 = 1582.32 nM T28887 C4DL0M 49847150 IC50 = 188 nM T28887 CC7Y9U 49850262 Ki = 96.2 nM T28887 C50PXU 49855444 IC50 = 2100 nM T28887 CE7D2J 49855568 IC50 = 11000 nM T28887 CFD9P3 49855569 IC50 = 19000 nM T28887 C1AU5N 49855758 IC50 = 31000 nM T28887 CIFK93 49855759 IC50 > 32000 nM T28887 CK48OJ 49855760 IC50 > 32000 nM T28887 CZI3M1 49855761 IC50 > 32000 nM T28887 CRPZ58 49855949 IC50 > 32000 nM T28887 CTU0K3 49855950 IC50 > 32000 nM T28887 CF85NL 49855951 IC50 > 32000 nM T28887 CF7YS9 49855952 IC50 = 7700 nM T28887 CJU38G 49855953 IC50 = 980 nM T28887 C5LZ4R 51351536 IC50 > 30000 nM T28887 C5LUD6 52950992 IC50 = 368 nM T28887 CAEP37 52950994 IC50 = 634 nM T28887 CC0VI7 52950996 IC50 = 481 nM T28887 CNKV26 52950998 IC50 = 1040 nM T28887 CLA8Y5 52951000 IC50 = 675 nM T28887 C13OGK 52951131 IC50 = 1280 nM T28887 C91YQC 52951133 IC50 = 1020 nM T28887 CYU0R2 52951254 IC50 = 192 nM T28887 C78BHS 52951255 IC50 = 201 nM T28887 C08BSF 52951359 IC50 = 147 nM T28887 CNC9V0 52951361 IC50 = 47 nM T28887 CSX0H2 52951363 IC50 = 68 nM T28887 C2IXJ1 52951365 IC50 = 1440 nM T28887 CSB58V 52951464 IC50 = 263 nM T28887 CZ9FU4 52951465 IC50 = 333 nM T28887 CSJ49T 52952070 IC50 = 502 nM T28887 CS1NL9 52952071 IC50 = 692 nM T28887 CB8RK1 52952072 IC50 = 759 nM T28887 C2KQ6A 52952387 IC50 = 514 nM T28887 CFB51H 52952488 IC50 = 103 nM T28887 C2UPR9 52952489 IC50 = 175 nM T28887 CLMX38 52952490 IC50 = 212 nM T28887 C6DAB7 52952491 IC50 = 139 nM T28887 CCH6W3 52952592 IC50 = 163 nM T28887 C86LAV 52952593 IC50 = 182 nM T28887 C1MRX4 52952594 IC50 = 104 nM T28887 CL9Y8K 52952595 IC50 = 141 nM T28887 CB79XD 52952596 IC50 = 164 nM T28887 CQ9UJ3 52952705 IC50 = 114 nM T28887 CIT60S 52952706 IC50 = 1720 nM T28887 C3AY8E 52952707 IC50 = 1020 nM T28887 CAZ78P 52952708 IC50 = 1920 nM T28887 C2YM1P 52952710 IC50 = 2140 nM T28887 CO7B2Y 53239053 IC50 = 260 nM T28887 CE43FC 53249967 IC50 = 200 nM T28887 C4NOS7 53309798 IC50 = 27600 nM T28887 C8SUQ5 53317424 IC50 > 30000 nM T28887 C7MO2J 53325871 IC50 = 1950 nM T28887 CVLE01 53345880 IC50 = 1860 nM T28887 CATU50 53357596 IC50 = 87 nM T28887 C5AQC7 53357597 IC50 = 86 nM T28887 CN0QR2 53357716 IC50 = 90 nM T28887 CVM4Q3 53357987 IC50 = 1090 nM T28887 C78GKN 53361474 IC50 = 17 nM T28887 CNB63X 53361475 IC50 = 651 nM T28887 C67VNG 53361476 IC50 = 76 nM T28887 CF3BK4 53361477 IC50 = 28 nM T28887 CX0U2Y 53362481 IC50 = 47100 nM T28887 CQD41A 53362535 IC50 = 36000 nM T28887 CD3HU6 53362593 IC50 = 707 nM T28887 CU2F1X 53362594 IC50 = 82 nM T28887 CC7L9E 53362595 IC50 = 147 nM T28887 CK74AM 53362596 IC50 = 487 nM T28887 CQ43VH 53363518 Ki = 55 nM T28887 C6Y2EV 53374826 IC50 = 954 nM T28887 C9WL1R 53387509 IC50 = 146 nM T28887 C6X5SA 53389591 IC50 = 21 nM T28887 CYQV72 54030066 IC50 = 15000 nM T28887 CTJ48R 54185618 IC50 = 753700 nM T28887 C0ZK7I 54576529 IC50 = 279.5 nM T28887 CTP2S1 54576530 IC50 = 267.85 nM T28887 CS8HY5 54576744 IC50 = 553.45 nM T28887 C5A7MU 54613496 IC50 = 282 nM T28887 CQ1EX7 54770442 IC50 = 1075.12 nM T28887 C7OJ4K 56602459 IC50 > 50000 nM T28887 CSY2L7 56602461 IC50 = 1200 nM T28887 CIO96M 56659403 IC50 > 100000 nM T28887 CX2ZF7 56659675 IC50 = 227 nM T28887 CP8RN3 56659683 IC50 = 63 nM T28887 C19MWJ 56659901 IC50 = 1310 nM T28887 CMW5G1 56659902 IC50 = 350 nM T28887 CEZ5I2 56659926 IC50 = 1930 nM T28887 CCI71R 56661654 IC50 = 960 nM T28887 C35QDT 56663143 IC50 = 660 nM T28887 C7R9TZ 56663191 IC50 = 102 nM T28887 C2JG3S 56663365 IC50 = 1070 nM T28887 CT1NL8 56663366 IC50 = 1440 nM T28887 CP47BX 56663394 IC50 = 1150 nM T28887 C8F9BM 56663395 IC50 = 720 nM T28887 CL18NI 56666337 IC50 > 100000 nM T28887 CIE5S9 56666802 IC50 = 2790 nM T28887 CB3DK0 56666803 IC50 = 140 nM T28887 C5C8BJ 56666805 IC50 = 690 nM T28887 CK3SP5 56670229 IC50 = 2520 nM T28887 C41YTB 56670231 IC50 = 10280 nM T28887 C9LC5Y 56673234 IC50 > 100000 nM T28887 CWH5N4 56673261 IC50 > 100000 nM T28887 C4IV8G 56673521 IC50 = 1180 nM T28887 C92JHM 56673753 IC50 = 760 nM T28887 CHD3I9 56673754 IC50 = 35 nM T28887 CV5WF9 56673770 IC50 = 1300 nM T28887 C6H3WB 56673771 IC50 = 600 nM T28887 C0ZJG3 56676500 IC50 = 30000 nM T28887 CZO78S 56676839 IC50 = 922 nM T28887 C5F8AS 56677091 IC50 = 2590 nM T28887 CES4U3 56677092 IC50 = 1190 nM T28887 CR1XM4 56677094 IC50 = 5900 nM T28887 COH9W3 56677096 IC50 = 1070 nM T28887 CRNW64 56677098 IC50 = 920 nM T28887 CU50WP 56678744 IC50 = 370 nM T28887 C7BNX6 56680155 IC50 = 151 nM T28887 CZ8K4S 56680156 IC50 = 213 nM T28887 C9G1MV 56680386 IC50 = 870 nM T28887 CS9IR1 56680418 IC50 = 4120 nM T28887 CFUT54 56682413 IC50 = 1000 nM T28887 CI2J9O 56683491 IC50 = 467 nM T28887 C9Q1NG 56683725 IC50 = 840 nM T28887 C7YL4Z 56683727 IC50 = 490 nM T28887 CXCI91 56683746 IC50 = 1900 nM T28887 C2ML5S 56837168 IC50 = 312 nM T28887 CXGV95 56929126 IC50 = 1600 nM T28887 CF81PW 56931564 IC50 = 4770 nM T28887 CCW89V 56932477 IC50 = 60.2 nM T28887 C7ABK4 56933019 IC50 = 470 nM T28887 CZ25SN 56935695 IC50 > 30000 nM T28887 C83UDV 56964457 IC50 = 220 nM T28887 CAW53S 57325672 IC50 = 4129 nM T28887 C9P8HJ 57325755 IC50 = 379 nM T28887 CG6Z2X 57326710 IC50 = 13000 nM T28887 C10DMC 57336560 Ki = 8400 nM T28887 C4LI0D 57521296 IC50 = 830 nM T28887 C8CQ7V 57523845 IC50 = 260 nM T28887 C4SK5V 57524018 IC50 = 590 nM T28887 CFHU47 57524021 IC50 = 410 nM T28887 CBZX29 57524107 IC50 = 76 nM T28887 C5LBS0 57524273 IC50 = 860 nM T28887 CVU30I 57524661 IC50 = 6250 nM T28887 CBM30D 57524665 IC50 = 150 nM T28887 C3VU1R 57524666 IC50 = 180 nM T28887 C3ZE4W 57524748 IC50 = 120 nM T28887 CJ68EZ 57524753 IC50 = 110 nM T28887 C4YNT9 57524833 IC50 = 120 nM T28887 C6A3CR 57524835 IC50 = 160 nM T28887 CTA82N 57524908 IC50 = 160 nM T28887 CXFJ46 57550498 IC50 = 4000 nM T28887 CA5Q6O 58147189 IC50 = 1300 nM T28887 C4DYC0 58147224 IC50 = 1300 nM T28887 CMP04X 58147302 IC50 = 890 nM T28887 C4V7FY 58191950 IC50 > 32000 nM T28887 CPCA29 58191961 IC50 = 590 nM T28887 C7HF1L 58191965 IC50 > 32000 nM T28887 CR4BX0 58191982 IC50 > 32000 nM T28887 C8V1NK 58191988 IC50 > 32000 nM T28887 C8LWY9 58191997 IC50 > 32000 nM T28887 C3IQ9B 58191999 IC50 > 32000 nM T28887 CQB69R 58192003 IC50 > 32000 nM T28887 CLD40J 58465708 IC50 = 3300 nM T28887 C1MB4Q 59323957 IC50 > 30000 nM T28887 CK6LX0 59454220 IC50 > 30000 nM T28887 C2SDN1 59454252 IC50 > 30000 nM T28887 CO6A2S 59585196 IC50 = 3300 nM T28887 CPZ5Q3 60148646 IC50 = 6700 nM T28887 CP2HK9 60148667 IC50 = 4800 nM T28887 C8ZL3J 60148690 IC50 = 1500 nM T28887 CK5N4E 60148693 IC50 = 360 nM T28887 C27DKW 60148711 IC50 = 1400 nM T28887 CS2E6C 60148712 IC50 = 5300 nM T28887 CPF50R 60148997 IC50 = 4300 nM T28887 CB7X2E 60151224 IC50 = 3550 nM T28887 CY05OU 60151225 IC50 > 10000 nM T28887 CWO8H0 60152596 IC50 > 10000 nM T28887 CXW14A 60164619 IC50 = 1584.89 nM T28887 CQ1U0P 60200243 IC50 = 2000 nM T28887 CZ18UT 67684770 IC50 > 1000000 nM T28887 CBN3L0 69950064 Ki = 7660 nM T28887 C6RFQ8 70676597 IC50 = 27 nM T28887 CQY1I6 70789579 Ki = 1330 nM T28887 C0I6VW 71139142 IC50 = 1570 nM T28887 C2ED7S 71139195 IC50 = 2780 nM T28887 CQO45N 71142065 IC50 = 6400 nM T28887 C8JK7A 71142076 IC50 = 2075 nM T28887 C50RGP 71142078 IC50 = 2858 nM T28887 CS1K8D 71142081 IC50 = 800 nM T28887 CG5FI7 71142082 IC50 = 6050 nM T28887 CFYV30 71142088 IC50 = 6751 nM T28887 C0ELR8 71142091 IC50 = 1660 nM T28887 CE4P1B 71142092 IC50 = 1465 nM T28887 CV8B4P 71142094 IC50 = 2402 nM T28887 CK6GL1 71142097 IC50 = 4283 nM T28887 C2RI8V 71142100 IC50 = 3105 nM T28887 C6L0JF 71142106 IC50 = 1868 nM T28887 C3D2KM 71142108 IC50 = 1482 nM T28887 CQU52J 71142109 IC50 = 2258 nM T28887 C2I9UX 71142126 IC50 = 1701 nM T28887 C25CUJ 71142127 IC50 = 2496 nM T28887 C96LSO 71142130 IC50 = 3303 nM T28887 C1KF3N 71142131 IC50 = 2533 nM T28887 CQ2E6U 71142135 IC50 = 2831 nM T28887 CA92XR 71449332 IC50 > 1000000 nM T28887 C8NZA0 71449818 IC50 = 67500 nM T28887 C63AHI 71449819 IC50 = 28000 nM T28887 CK2AT8 71451145 IC50 = 825100 nM T28887 C5NYF7 71451146 IC50 = 47200 nM T28887 CW06TJ 71451147 IC50 = 3600 nM T28887 C7UIS9 71452970 IC50 > 1000000 nM T28887 CC1B0Z 71452971 IC50 > 1000000 nM T28887 CNMP23 71452972 IC50 = 871500 nM T28887 CIP9J5 71452973 IC50 > 1000000 nM T28887 CUZ9S0 71452974 IC50 = 102300 nM T28887 C71TWC 71452975 IC50 = 52500 nM T28887 CGE27K 71454723 IC50 = 36900 nM T28887 C4EJX2 71456472 IC50 = 5800 nM T28887 C6B2HJ 71456958 IC50 = 750 nM T28887 CUY95O 71456963 IC50 = 47800 nM T28887 C1JI6W 71458326 IC50 > 1000000 nM T28887 C8ZR2I 71458327 IC50 = 9300 nM T28887 CV2J5Y 71458328 IC50 = 30700 nM T28887 C29YHS 71458330 IC50 = 27800 nM T28887 C3NL2S 71458833 IC50 = 53200 nM T28887 CKV4Q6 71460169 IC50 = 385600 nM T28887 CYF62U 71460170 IC50 = 120900 nM T28887 C3LFX2 71460171 IC50 > 1000000 nM T28887 CDRO30 71460172 IC50 = 42400 nM T28887 C6WN3A 71460173 IC50 = 14400 nM T28887 CX7W4A 71461879 IC50 > 1000000 nM T28887 CKXO81 71461880 IC50 = 961800 nM T28887 CI4M8V 71461881 IC50 = 253400 nM T28887 CHD70Q 71461882 IC50 = 9500 nM T28887 C7MLC8 71461883 IC50 = 82500 nM T28887 CH2O7D 71462353 IC50 = 42600 nM T28887 C0CX7P 71476624 Ki = 2.27 nM T28887 C6QPH1 71476625 Ki = 122.7 nM T28887 C3JLD4 71476626 Ki = 2.38 nM T28887 C3OH6T 71476627 Ki = 266.3 nM T28887 CFQ2N9 71520536 IC50 = 11170 nM T28887 C0LWJ6 71520631 IC50 = 1043 nM T28887 CO28HI 71520716 IC50 = 833 nM T28887 CVA5Q7 71520717 IC50 = 1278 nM T28887 C6KBD4 71534512 IC50 = 2570 nM T28887 CT51EW 71534810 IC50 = 360 nM T28887 C7QN3O 71534812 IC50 = 135 nM T28887 C8M3HU 71537640 IC50 = 2040 nM T28887 C2QML7 71537641 IC50 = 40 nM T28887 CZJX53 71537927 IC50 = 2230 nM T28887 CU0ZE6 71537928 IC50 = 281 nM T28887 CH9FS7 71537929 IC50 = 17 nM T28887 CTW95A 71537931 IC50 = 122 nM T28887 C3C0RO 71538475 IC50 = 202 nM T28887 CIA28E 71538746 IC50 = 416 nM T28887 CFCV26 71538748 IC50 = 9 nM T28887 CY2T1Q 71538749 IC50 = 23 nM T28887 C4A6VJ 71538750 IC50 = 61 nM T28887 CG72NC 71538751 IC50 = 310 nM T28887 CDW81Y 71574856 IC50 = 20910 nM T28887 CX01BJ 71574948 IC50 = 1330 nM T28887 CO8YU7 71574949 IC50 = 1950 nM T28887 CKR6U8 71583101 IC50 = 2800 nM T28887 CBZ5S9 71583103 IC50 = 1700 nM T28887 C3PSJ9 71583105 IC50 = 900 nM T28887 C21GHR 71624738 IC50 = 6000 nM T28887 CBN92Q 71625222 IC50 = 1726 nM T28887 CCQ0U1 71625341 IC50 = 2599 nM T28887 CD09SV 71625344 IC50 = 1046 nM T28887 C7HG0K 71655802 IC50 = 1090 nM T28887 CPJ4V7 71680913 IC50 = 120 nM T28887 C9X8KM 71680914 IC50 = 420 nM T28887 C4W2MA 71680915 IC50 = 210 nM T28887 C3KO9V 71680916 IC50 = 110 nM T28887 CN4X5O 71680917 IC50 = 14000 nM T28887 CWAM13 71680918 IC50 = 1700 nM T28887 CI9G3B 71681069 IC50 = 37 nM T28887 C5WZV9 71720123 IC50 = 1907 nM T28887 CIR56T 71721558 IC50 > 100000 nM T28887 CCD18W 71721946 IC50 > 30000 nM T28887 CFUC24 71722010 IC50 = 420.9 nM T28887 CEG67K 71723449 IC50 = 130 nM T28887 C0P8CH 71748076 IC50 = 173 nM T28887 CU4X2F 71761851 IC50 = 11000 nM T28887 C7SK3L 71761852 IC50 = 5000 nM T28887 CI2NH1 71761853 IC50 = 4000 nM T28887 CORB04 71762088 IC50 = 450 nM T28887 CYG6O7 71762089 IC50 = 20000 nM T28887 CTSK68 71811225 IC50 = 1750 nM T28887 C1K6OW 71811226 IC50 = 1270 nM T28887 CU3N9R 71811227 IC50 = 3880 nM T28887 CS2L4B 71811228 IC50 = 1590 nM T28887 CL4DT9 71811229 IC50 = 600 nM T28887 CK6DB4 71811230 IC50 = 1330 nM T28887 CHR8V0 71811259 IC50 = 1180 nM T28887 CVL54T 71811261 IC50 = 282 nM T28887 CZR93K 71811262 IC50 = 891 nM T28887 CM8BE4 71811290 IC50 = 594 nM T28887 C0MV3O 71811291 IC50 = 1060 nM T28887 C7UYD4 71811292 IC50 = 609 nM T28887 C7XL3N 71811293 IC50 = 420 nM T28887 C4HBC5 71811294 IC50 = 1400 nM T28887 CTA26S 71811295 IC50 = 766 nM T28887 C9GHU8 71818097 IC50 = 1400 nM T28887 CAW2Q1 71818098 IC50 = 2300 nM T28887 CE89AK 71818242 IC50 > 20000 nM T28887 C8M3IX 71818243 IC50 > 20000 nM T28887 CKP5J7 71818244 IC50 = 5160 nM T28887 CT7L6G 72163687 Ki = 186.3 nM T28887 CKE9D3 72163688 Ki = 123.65 nM T28887 CI9H6L 72164895 IC50 = 2311 nM T28887 CH68XV 72188554 IC50 = 1970 nM T28887 CS5UL7 72195322 IC50 = 2984 nM T28887 C3WQV2 72375562 IC50 = 1200 nM T28887 C1A4YW 72545684 IC50 = 1460 nM T28887 CJR6C9 72734542 IC50 = 820 nM T28887 CV09DJ 72734543 IC50 = 5000 nM T28887 CS6LW0 72946640 IC50 = 97 nM T28887 CXM37Z 72946641 IC50 = 161 nM T28887 CQA16N 72946833 IC50 = 137 nM T28887 CNR7Z2 72946834 IC50 = 251 nM T28887 C12JYS 72946835 IC50 = 118 nM T28887 C5Y9XH 72946836 IC50 = 123 nM T28887 CVZR94 72946837 IC50 = 2130 nM T28887 C8-AUG 72946838 IC50 = 131 nM T28887 CHQ39Y 72947043 IC50 = 137 nM T28887 CCST90 72947044 IC50 = 52 nM T28887 C7J3RH 72947045 IC50 = 156 nM T28887 CK10LZ 73292342 IC50 = 1880 nM T28887 CX3W1T 73333311 IC50 = 690 nM T28887 C21XQI 73345596 IC50 = 230 nM T28887 CDG47J 73346009 IC50 > 20000 nM T28887 C6H7IJ 73346010 IC50 > 20000 nM T28887 CD0WU2 73346011 IC50 > 20000 nM T28887 COBJ19 73347538 IC50 > 20000 nM T28887 C92HFB 73349064 IC50 > 20000 nM T28887 C68LBO 73349131 IC50 = 2580 nM T28887 CAS8E2 73352138 IC50 > 20000 nM T28887 CSP58Q 73353181 IC50 = 370 nM T28887 CH6Z2L 73353182 IC50 = 780 nM T28887 C0C2QO 73353595 IC50 > 20000 nM T28887 C59WMZ 73353596 IC50 > 20000 nM T28887 C1UDF8 73353597 IC50 > 20000 nM T28887 CUD02X 73355098 IC50 = 410 nM T28887 CXK86S 73355189 IC50 = 2660 nM T28887 CNC6Q5 73505594 IC50 = 390 nM T28887 CZB6G7 73776472 IC50 = 2000.8 nM T28887 C3UC9H 73891099 IC50 = 1600 nM T28887 CP30HW 76308051 IC50 = 90 nM T28887 CUX1G5 76311607 IC50 = 8.5 nM T28887 CX3EY4 76311608 IC50 = 9.5 nM T28887 C3YH9X 76314009 IC50 = 1377 nM T28887 CCS3A7 76315181 IC50 = 95 nM T28887 CPX70Y 76315182 IC50 = 15 nM T28887 CYSV86 76315183 IC50 = 5 nM T28887 C3D2HY 76315214 IC50 = 600 nM T28887 CG7R8F 76318826 IC50 = 460 nM T28887 CQ83VF 76318827 IC50 = 8 nM T28887 CT48EH 76318828 IC50 = 4.5 nM T28887 C9ID1J 76318869 IC50 = 2000 nM T28887 CK5SF2 76322485 IC50 = 71.4 nM T28887 CH76MT 76322486 IC50 = 153 nM T28887 CFSY27 76322487 IC50 = 45 nM T28887 C1QMH9 76322488 IC50 = 45 nM T28887 C1F2CU 76322523 IC50 = 35 nM T28887 C7C8JK 76322524 IC50 = 100 nM T28887 CM6H9C 76324878 IC50 = 870 nM T28887 C3OF6T 76326087 IC50 = 600 nM T28887 CZ7HA9 76326118 IC50 = 17000 nM T28887 CAJ3F6 76329682 IC50 = 20 nM T28887 CY3XA9 76329683 IC50 = 135 nM T28887 CPDV98 76329684 IC50 = 2 nM T28887 CPX4F1 76329718 IC50 = 25 nM T28887 CL4JQ3 76331862 IC50 = 1410 nM T28887 C8RXP4 76333350 IC50 = 4 nM T28887 CBM6U8 76333386 IC50 = 6 nM T28887 CJW53Q 76333387 IC50 = 60 nM T28887 C08CPW 76335428 IC50 = 31.6 nM T28887 C7JQU3 76335755 IC50 = 917 nM T28887 CKI74A 76853213 IC50 = 0.8 nM T28887 CCR7L2 76853289 IC50 = 150 nM T28887 C96LMJ 78323868 IC50 = 150 nM T28887 C5IAU4 78323870 IC50 = 200 nM T28887 CJ6Z0X 78324068 IC50 = 10 nM T28887 C25ETN 78324161 IC50 = 320 nM T28887 C3U0KE 81689842 IC50 = 9100 nM T28887 CG5ZD9 86291495 IC50 = 6 nM T28887 C61VCD 86294741 IC50 = 980 nM T28887 CBWV30 86294747 IC50 = 1200 nM T28887 C06YBD 86302594 IC50 = 1760 nM T28887 C3EM7H 86581004 IC50 = 53 nM T28887 C7UK3Y 86581005 IC50 = 55 nM T28887 CY64UM 86581152 IC50 = 94 nM T28887 CY5V7C 86581153 IC50 = 33 nM T28887 C1HE8I 86581432 IC50 = 200 nM T28887 CZM07I 86581434 IC50 = 49 nM T28887 C8ZQG9 86581435 IC50 = 24 nM T28887 C6M9PL 86765212 IC50 = 1390 nM T28887 CS5I4Y 87261507 IC50 = 150 nM T28887 C5JIT0 87618609 IC50 > 32000 nM T28887 CRQO37 88005144 IC50 > 32000 nM T28887 CRAX13 88849486 IC50 = 760 nM T28887 CD3X6M 88849490 IC50 = 210 nM T28887 CYW51P 90654946 IC50 = 2910 nM T28887 CJH1S6 90654947 IC50 = 30600 nM T28887 CSR56C 90655296 IC50 = 717 nM T28887 CSDO81 90664458 Ki = 48 nM T28887 C67UHD 91619090 IC50 = 38500 nM T28887 C6JZT7 91619093 IC50 = 41900 nM T28887 C5M9AK 91667421 IC50 = 1491 nM T28887 CJO6T1 91810840 IC50 = 400 nM T28887 CYJ12Q 91884636 IC50 = 281 nM T28887 C34WIG 92045024 IC50 = 80 nM T28887 CN5KS8 92135978 IC50 = 171.5 nM T28887 C9OC0F 101882265 IC50 = 30 nM T28887 CDV40P 101882454 IC50 = 290 nM T28887 C0M1NK 101882456 IC50 = 460 nM T28887 CPUJ32 101882458 IC50 = 420 nM T28887 C7Q6ID 101884982 IC50 = 59 nM T28887 CR46PQ 101884983 IC50 = 107 nM T28887 CRZ83C 101884989 IC50 = 8100 nM T28887 CT7Z8F 102514716 IC50 = 1536 nM T28887 CS2UL0 117829456 IC50 = 80 nM T28887 C7L4OT 117829461 IC50 = 59 nM T28887 C50VUN 117829462 IC50 = 72 nM T28887 C0OX4M 118613748 IC50 = 540 nM T28887 C46TFD 118613757 IC50 = 790 nM T28887 CSU52M 118656852 IC50 = 2400 nM T28887 CB6AJ9 118656853 IC50 = 1900 nM T28887 C45UYG 118709095 IC50 = 28000 nM T28887 C1JFZ7 118714371 IC50 = 2515 nM T28887 CXF0U3 118714375 IC50 = 4918 nM T28887 C2M5OR 118714376 IC50 = 1024 nM T28887 CY4GN9 118714377 IC50 = 5238 nM T28887 C96XGO 118715268 IC50 = 390 nM T28887 CM5QT7 118719376 Ki = 6000 nM T28887 C09OGH 118719378 Ki = 3000 nM T28887 C8U6YR 118719381 Ki = 4300 nM T28887 CY0J4D 118719383 Ki = 4500 nM T28887 CCYU59 118719817 IC50 = 316 nM T28887 CUI51W 118720529 IC50 = 87.4 nM T28887 CMV2W9 118721625 IC50 = 62 nM T28887 CF5TO3 118721859 IC50 = 545 nM T28887 CK97TZ 118721860 IC50 = 106 nM T28887 CYV30O 118721861 IC50 = 106 nM T28887 C5WYI1 118721862 IC50 = 99 nM T28887 CSMW25 118721863 IC50 = 2330 nM T28887 C5B1KM 118721864 IC50 = 450 nM T28887 CG8LZ0 118721865 IC50 = 373 nM T28887 CPCN23 118721866 IC50 = 904 nM T28887 CM0A9U 118721867 IC50 = 246 nM T28887 CN47HE 118733259 IC50 = 8200 nM T28887 CJLN15 118733260 IC50 = 4920 nM T28887 CU8T7G 118733373 IC50 = 22400 nM T28887 C6OEU2 118733374 IC50 = 180 nM T28887 CW5JY8 118733375 IC50 = 590 nM T28887 C16OUT 118735146 IC50 > 10000 nM T28887 CZRV81 118735147 IC50 > 10000 nM T28887 CFE4D0 118735148 IC50 > 10000 nM T28887 C97NHV 118735149 IC50 > 10000 nM T28887 CQ0FJ3 118735150 IC50 > 10000 nM T28887 CD4J8E 118735151 IC50 > 10000 nM T28887 C7UE8T 118735152 IC50 > 10000 nM T28887 CS6WO5 118735153 IC50 > 10000 nM T28887 C4XZ3C 118735154 IC50 > 10000 nM T28887 CRL6V4 118735155 IC50 > 10000 nM T28887 CI8G4X 118737400 IC50 = 610 nM T28887 C2F8TQ 118737455 IC50 = 343 nM T28887 C1T6WZ 118738004 IC50 > 10000 nM T28887 CZ61KV 118753026 IC50 = 920 nM T28887 CFI23Y 118753027 IC50 = 23000 nM T28887 C75LTK 118753189 IC50 = 6800 nM T28887 CM3FB8 118796366 IC50 = 582 nM T28887 C8DVP1 118868599 Ki = 1678 nM T28887 C9G4LD 118868621 Ki = 720 nM T28887 CQT5I6 118868656 Ki = 1540 nM T28887 CE3PD1 118868670 Ki > 40000 nM T28887 C5L8QM 118884518 IC50 = 747 nM T28887 CV0E3L 118884590 Ki = 528 nM T28887 CME8R7 118884591 Ki = 427 nM T28887 C4XJ7F 118884592 Ki = 205 nM T28887 CP5TE9 118884676 Ki = 701 nM T28887 CVTL89 118884679 Ki = 299 nM T28887 CB84TO 121278998 IC50 = 57 nM T28887 C9S5OK 121279020 IC50 = 830 nM T28887 CIA40K 121472983 IC50 = 2100 nM T28887 CL3M2F 121499152 IC50 > 33330 nM T28887 C93JAV 122177622 Ki = 250 nM T28887 C5HJ0C 122177623 IC50 > 10000 nM T28887 CSU97K 122177957 IC50 = 2.5 nM T28887 CR8WL1 122180003 IC50 = 7650 nM T28887 C0H9WU 122181882 IC50 = 101.8 nM T28887 C9V6XI 122186483 IC50 = 5500 nM T28887 CU74JP 122186484 IC50 = 14300 nM T28887 C7M2EU 122186485 IC50 = 9500 nM T28887 CCG1Z2 122186543 IC50 = 112000 nM T28887 CI32QY 122186544 IC50 = 88000 nM T28887 CBN3P1 122186553 IC50 = 173000 nM T28887 CP83NA 122186554 IC50 = 8100 nM T28887 C28JVO 122192004 IC50 = 2550 nM T28887 CF2D8U 122192005 IC50 > 10000 nM T28887 CV8YH0 122193364 IC50 = 14300 nM T28887 C1CI0Z 122193365 IC50 = 8010 nM T28887 C32LTK 122193367 IC50 = 1800 nM T28887 CE04LR 122193368 IC50 = 1620 nM T28887 CW1HK5 122195536 IC50 = 5.2 nM T28887 C5W8OZ 122376192 IC50 = 1810 nM T28887 CL0X8K 122550124 IC50 > 1000 nM T28887 C24QLO 122550126 IC50 = 1510 nM T28887 CNKM78 122550129 IC50 = 2457 nM T28887 CL31AN 122550132 IC50 = 1422 nM T28887 CJM9X5 122550134 IC50 = 1326 nM T28887 CHS4F7 122550135 IC50 = 1058 nM T28887 CB8J6A 122550165 IC50 > 1000 nM T28887 CZ6TC9 122550171 IC50 > 1000 nM T28887 CX87LD 122550174 IC50 = 5189 nM T28887 C3V5ND 122550211 IC50 = 3398 nM T28887 C64OME 122550212 IC50 = 1465 nM T28887 C8PM6C 122550213 IC50 = 1531 nM T28887 CAXY60 122550234 IC50 = 1181 nM T28887 CAOH68 122550235 IC50 = 1698 nM T28887 CR38WT 122550251 IC50 > 1000 nM T28887 CX61TL 122550293 IC50 > 1000 nM T28887 C63EYP 122601008 IC50 = 230 nM T28887 CCN03D 122601010 IC50 = 2200 nM T28887 CZC01M 122601076 IC50 = 110 nM T28887 CZE35C 122648343 IC50 = 92.92 nM T28887 C54RNT 122648367 IC50 = 24 nM T28887 C1UVI7 122648600 IC50 = 217 nM T28887 CMX59K 122648648 IC50 = 22 nM T28887 CVZ64I 122648649 IC50 = 11 nM T28887 CZ67DK 126738293 IC50 = 12000 nM T28887 CVFI87 127025051 IC50 = 2000 nM T28887 CQ39UE 127025078 IC50 = 33890 nM T28887 CE4CI8 127025178 IC50 > 10000 nM T28887 CM38EU 127025541 IC50 = 4200 nM T28887 CY5T9P 127025646 IC50 = 130 nM T28887 CKJ6L8 127025647 IC50 = 54 nM T28887 CXVC21 127025656 IC50 = 30760 nM T28887 CWB73C 127025940 IC50 = 20040 nM T28887 C6D2IJ 127026516 IC50 = 2010 nM T28887 CNH5P8 127026863 IC50 = 35000 nM T28887 CSJ18X 127027150 IC50 = 29080 nM T28887 CA58GI 127027171 IC50 = 14370 nM T28887 CBT4S5 127027172 IC50 = 20240 nM T28887 C3UED2 127027173 IC50 = 43350 nM T28887 CUSY71 127027174 IC50 = 50940 nM T28887 C2OIE1 127027175 IC50 = 26160 nM T28887 COU4I9 127027458 IC50 = 2700 nM T28887 CC0WJ2 127027462 IC50 = 8130 nM T28887 CSZL73 127027477 IC50 = 36360 nM T28887 CY3P7V 127027483 IC50 = 10080 nM T28887 C68TYH 127027490 IC50 > 30000 nM T28887 C8BA3S 127027767 IC50 = 1440 nM T28887 CD4T1B 127027794 IC50 = 12860 nM T28887 CG7Q3V 127027808 IC50 > 30000 nM T28887 C6JUF9 127027813 IC50 > 30000 nM T28887 CG8NU7 127027995 IC50 > 10000 nM T28887 CZ7C3D 127028030 IC50 = 4.6 nM T28887 CL7EN6 127028391 IC50 = 27330 nM T28887 CW04XE 127028723 IC50 = 12120 nM T28887 CV07OM 127028943 IC50 > 10000 nM T28887 CV9I8D 127030313 IC50 = 580 nM T28887 CN6K5P 127030500 IC50 = 1987 nM T28887 CCNK89 127030846 IC50 > 1000 nM T28887 CI8WG4 127031734 IC50 = 6190 nM T28887 C40HQA 127031756 IC50 = 2974 nM T28887 C9Q1WD 127031757 IC50 = 1003 nM T28887 CD1TP7 127034929 IC50 = 1190 nM T28887 CU1M3B 127034930 IC50 = 2450 nM T28887 C4SI0Q 127034947 IC50 = 2240 nM T28887 CMS1F6 127034948 IC50 = 3210 nM T28887 C3VB0I 127034949 IC50 = 2030 nM T28887 CQC2F9 127035098 IC50 = 3230 nM T28887 CBP64A 127035107 IC50 = 310 nM T28887 CAXL98 127035256 IC50 = 2850 nM T28887 CBJG94 127035257 IC50 > 10000 nM T28887 C29AJN 127035766 IC50 = 1500 nM T28887 CSJ32V 127039213 IC50 = 3130 nM T28887 C18FSM 127039340 IC50 = 160 nM T28887 CIO0G3 127039341 IC50 = 200 nM T28887 C12NJF 127039347 IC50 = 570 nM T28887 C69IXG 127041845 IC50 = 430 nM T28887 CO72YC 127045674 IC50 = 30.3 nM T28887 CTG0U3 127045675 IC50 = 26.1 nM T28887 CD42EQ 127045676 IC50 = 77.1 nM T28887 C9K0TN 127045677 IC50 = 239.7 nM T28887 CK51QO 127045678 IC50 = 548.3 nM T28887 CI8GB3 127046027 IC50 = 104.3 nM T28887 C0HQZ3 127046055 IC50 = 830 nM T28887 CG13WB 127046056 IC50 = 2190 nM T28887 CIQA39 127046057 IC50 = 204 nM T28887 CFP10C 127046594 IC50 = 143.4 nM T28887 CC89WM 127046659 IC50 = 342.2 nM T28887 CR61BE 127046852 IC50 = 1184 nM T28887 CXJM94 127046853 IC50 = 148.7 nM T28887 C42VYT 127046854 IC50 = 23.9 nM T28887 CR6AH4 127046855 IC50 = 19.8 nM T28887 CM76WI 127046917 IC50 = 191.4 nM T28887 CQ8LT6 127047324 IC50 = 292 nM T28887 CJ7YR6 127047335 IC50 = 235.6 nM T28887 CB0O4H 127047412 IC50 = 438.4 nM T28887 C5OH2V 127047413 IC50 = 512.2 nM T28887 CEUB27 127047550 IC50 = 214.4 nM T28887 CU1M3Q 127047551 IC50 = 448.6 nM T28887 CKH4S0 127047552 IC50 = 1080 nM T28887 C7TV8A 127047636 IC50 = 211.16 nM T28887 C4N2BY 127047651 IC50 = 88.3 nM T28887 C5SW8E 127047652 IC50 = 317.8 nM T28887 CE1K8N 127047653 IC50 = 120 nM T28887 C2KB3W 127048062 IC50 = 29 nM T28887 CB8HR2 129104138 IC50 = 130 nM T28887 CCH65A 129104183 IC50 = 1100 nM T28887 CFH8Q4 129104227 IC50 = 1800 nM T28887 C6HM5P 129104349 IC50 = 13000 nM T28887 CZTF90 129104374 IC50 = 21000 nM T28887 CUJ2P5 129104402 IC50 = 6700 nM T28887 CY3I6X 129104426 IC50 = 540 nM T28887 CA9EV6 130205513 IC50 = 240 nM T28887 C8KRX0 130205516 IC50 = 340 nM T28887 CJ7CQ5 130205526 IC50 = 60 nM T28887 CUHY85 130205779 IC50 = 6200 nM T28887 CGT6B0 130238385 Ki = 40.4 nM T28887 CMWV13 130238420 Ki = 124 nM T28887 C0GH4T 130238474 Ki = 93.3 nM T28887 C9ERM5 130238475 Ki = 13.09 nM T28887 C8IEV4 130258911 IC50 = 168 nM T28887 CHVF85 132022730 IC50 = 1400 nM T28887 C6OXE3 132134663 IC50 = 740 nM T28887 C6X3HG 132145728 IC50 = 636 nM T28887 C8O9DP 132157820 IC50 = 1190 nM T28887 C2N5JD 132279660 IC50 = 98 nM T28887 C4L6UZ 132547258 IC50 = 345 nM T28887 CGBR54 132547259 IC50 = 412 nM T28887 CW4MP2 132547260 IC50 = 109 nM T28887 C1YO2Z 132547261 IC50 = 135 nM T28887 C0Y2TP 132585192 IC50 = 2750 nM T28887 C4KE3N 132938351 IC50 = 211 nM T28887 C4UAN3 134129876 IC50 = 520 nM T28887 C25EVA 134129883 IC50 = 116 nM T28887 CWRH43 134129994 IC50 = 544 nM T28887 CK2TM6 134130010 IC50 = 226 nM T28887 CYW6H1 134130165 IC50 = 697 nM T28887 C8CY7S 134131006 IC50 = 707 nM T28887 CQ7SN8 134131102 IC50 = 989 nM T28887 CYCS54 134131113 IC50 = 345 nM T28887 CQO23I 134131456 IC50 = 394 nM T28887 CHZ8A3 134131564 IC50 = 672 nM T28887 CN8L9J 134136160 IC50 = 3100 nM T28887 C6URA0 134139607 IC50 = 116 nM T28887 C08YTI 134140697 IC50 = 200 nM T28887 C3D1UF 134143133 IC50 = 139 nM T28887 CUA26W 134143927 IC50 = 1300 nM T28887 COI36H 134144171 IC50 = 134 nM T28887 CYK6E2 134147070 IC50 = 142 nM T28887 C1NA7J 134148049 IC50 = 135 nM T28887 CKCB54 134152269 IC50 = 153 nM T28887 CTBN42 134154194 IC50 = 121 nM T28887 C2E8MV 134154228 IC50 = 130 nM T28887 C4S2FY 134155619 IC50 = 155 nM T28887 CP89YB 134156598 IC50 = 127 nM T28887 C38DIF 134156853 IC50 = 2000 nM T28887 CU4I0P 134158029 IC50 = 710 nM T28887 C9DSR3 134159676 IC50 = 260 nM T28887 CZV43J 134283792 IC50 = 74 nM T28887 C62WXO 134283796 IC50 = 150 nM T28887 CO7K3N 134283799 IC50 = 130 nM T28887 CBQ17L 134283800 IC50 = 27 nM T28887 C1Y4TA 134283810 IC50 = 79 nM T28887 CV2YF7 134283813 IC50 = 57 nM T28887 C05FVT 134492522 IC50 = 5600 nM T28887 CWJ7D1 134611695 IC50 = 3100 nM T28887 CML7O0 134822021 IC50 = 155 nM T28887 C52IBY 134823859 IC50 = 530 nM T28887 C14FWK 135348858 IC50 = 1230 nM T28887 CS1V6A 135367138 IC50 = 520 nM T28887 CVO59N 135367789 IC50 = 2700 nM T28887 CDY18W 135407493 IC50 > 100000 nM T28887 CW2I4R 135412048 IC50 > 100000 nM T28887 C7U0AV 135412194 IC50 > 100000 nM T28887 CS54TL 135437514 IC50 > 100000 nM T28887 C36MUC 135441620 IC50 > 100000 nM T28887 CRB8M1 135444536 IC50 > 100000 nM T28887 CX5D6J 135446479 IC50 = 23900 nM T28887 C1TOK2 135449197 IC50 > 100000 nM T28887 CW25GL 135462117 IC50 > 100000 nM T28887 CCL28F 135473106 IC50 > 100000 nM T28887 CYA60G 135497781 IC50 > 100000 nM T28887 C01EZF 135567459 IC50 = 746 nM T28887 C6GYM1 135567460 IC50 = 2200 nM T28887 CP2V6K 135860584 IC50 = 33670 nM T28887 C8X5LO 135928012 Ki = 50 nM T28887 CI2YE8 135928628 IC50 > 100000 nM T28887 C50NIS 136025837 IC50 > 100000 nM T28887 C4OS0V 136025842 IC50 > 100000 nM T28887 CX7Z5B 136025843 IC50 > 100000 nM T28887 CB8EM9 136025984 IC50 > 100000 nM T28887 C49MUG 136025986 IC50 > 100000 nM T28887 C0OLS8 136030779 IC50 = 350 nM T28887 CIA7R4 136030780 IC50 = 180 nM T28887 C24LKN 136030781 IC50 = 100 nM T28887 C1MGP6 136033554 IC50 = 15700 nM T28887 CH7Y3C 136086920 IC50 > 100000 nM T28887 C3VDL5 136086921 IC50 > 100000 nM T28887 C9GOB5 136086922 IC50 > 100000 nM T28887 CE3ZL7 136086923 IC50 > 100000 nM T28887 CJZ5F3 136086924 IC50 > 100000 nM T28887 CT19ND 136110961 IC50 = 25200 nM T28887 CY9U0E 136173089 IC50 = 610 nM T28887 C19VDS 136237971 IC50 = 23500 nM T28887 CBS97C 136239447 IC50 = 4100 nM T28887 CT2MI6 136239448 IC50 = 15000 nM T28887 CE2F9G 136244081 IC50 = 10700 nM T28887 C9CH7S 136244085 IC50 = 34900 nM T28887 C5J2AX 136244086 IC50 = 12700 nM T28887 C46CYT 136244087 IC50 = 14900 nM T28887 CXY1L5 136244088 IC50 = 12600 nM T28887 CRPN39 136645466 IC50 > 10000 nM T28887 CE6QK0 137125258 IC50 = 179000 nM T28887 CAW80Q 137125259 IC50 = 63000 nM T28887 CP5NM4 137125260 IC50 = 29200 nM T28887 C5CKZ8 137125261 IC50 = 80700 nM T28887 C1ROQ9 137125262 IC50 = 113000 nM T28887 CL29YN 137125263 IC50 = 88000 nM T28887 C5OY8K 137125264 IC50 = 33900 nM T28887 C0YGR6 137125265 IC50 = 52200 nM T28887 CMYG96 137125266 IC50 = 82100 nM T28887 CI78CK 137125267 IC50 = 83300 nM T28887 CD62KP 137125268 IC50 = 53500 nM T28887 CE8NM5 137125269 IC50 = 111000 nM T28887 CM1N3O 137226378 IC50 = 61420 nM T28887 CWM6Z2 137376574 Ki = 761 nM T28887 C3LUJ0 137487429 IC50 = 2890 nM T28887 C67EFJ 137628684 IC50 = 1.28 nM T28887 CX0PH5 137628685 IC50 > 1000 nM T28887 CG23FD 137631444 IC50 > 30000 nM T28887 C9UQD2 137631509 IC50 > 30000 nM T28887 CP0JL9 137631552 IC50 > 30000 nM T28887 CI7H8W 137631674 IC50 = 114 nM T28887 CP0BN3 137631704 Ki > 50000 nM T28887 C31MPL 137631726 IC50 = 1540 nM T28887 CJ9GD5 137631769 IC50 > 30000 nM T28887 CQ54WK 137631915 IC50 > 30000 nM T28887 CD1L0I 137632135 IC50 > 30000 nM T28887 C1N8TU 137632249 Ki = 294 nM T28887 C6A4GK 137632422 IC50 > 30000 nM T28887 CQ4BK9 137632561 IC50 > 30000 nM T28887 CVB93K 137632723 IC50 = 24750 nM T28887 CV8A5X 137632749 IC50 = 167 nM T28887 C9RWF1 137632979 IC50 > 30000 nM T28887 CI2G7B 137633049 IC50 > 30000 nM T28887 CMU42D 137633092 IC50 > 30000 nM T28887 CY08AM 137633123 IC50 > 30000 nM T28887 C84MIY 137633138 IC50 > 100000 nM T28887 CZY46A 137633389 IC50 = 254 nM T28887 C1HL3I 137633415 IC50 > 30000 nM T28887 C73PDL 137634086 IC50 > 100000 nM T28887 C1V8QE 137634156 IC50 = 398.11 nM T28887 C2M9NR 137634298 IC50 = 119 nM T28887 C8G4KJ 137634562 IC50 > 30000 nM T28887 CJ76DN 137634596 IC50 > 30000 nM T28887 C7U1CE 137634604 IC50 > 30000 nM T28887 C31DRY 137634704 IC50 = 481 nM T28887 C90TSR 137634950 IC50 > 30000 nM T28887 CZ1FK2 137635119 IC50 = 557.3 nM T28887 CHA4E3 137635225 IC50 > 30000 nM T28887 C6JVG9 137635398 IC50 = 469 nM T28887 CBMN61 137635405 IC50 > 30000 nM T28887 CAWZ25 137635575 IC50 > 100 nM T28887 CZ29MT 137635651 IC50 > 30000 nM T28887 C7N5BG 137635855 IC50 > 30000 nM T28887 C2MB4U 137636234 IC50 > 30000 nM T28887 CA2S3J 137636481 IC50 > 30000 nM T28887 C5GCO8 137636604 IC50 > 30000 nM T28887 CSY3E1 137636623 IC50 = 72 nM T28887 C72SBN 137636632 IC50 > 30000 nM T28887 C9THE6 137636891 IC50 > 30000 nM T28887 CF3E8T 137637310 IC50 > 30000 nM T28887 C6MVX0 137637661 IC50 = 22390 nM T28887 C3H2GO 137637718 IC50 > 30000 nM T28887 CSH08B 137637787 IC50 > 30000 nM T28887 CEI0W2 137637915 IC50 = 420 nM T28887 CMU93I 137637990 IC50 > 30000 nM T28887 CMD89K 137638151 IC50 > 30000 nM T28887 CQ3DR6 137638257 IC50 > 30000 nM T28887 CO9UY1 137638342 IC50 > 30000 nM T28887 C3RC2O 137638626 IC50 > 30000 nM T28887 CEMX30 137638687 IC50 > 30000 nM T28887 CTUL07 137638741 IC50 > 100 nM T28887 CTG6X0 137638748 IC50 > 30000 nM T28887 CX8Q4R 137638837 Ki = 721 nM T28887 CZU31H 137638926 IC50 = 3300 nM T28887 CQ86FE 137638947 IC50 > 30000 nM T28887 C7IJC2 137639014 IC50 = 20280 nM T28887 C69IOZ 137639088 IC50 = 1080 nM T28887 C2DIM1 137639536 IC50 = 19830 nM T28887 CW4DJ8 137639563 IC50 > 30000 nM T28887 CS9A6C 137639566 IC50 > 30000 nM T28887 CMI6Z0 137639764 IC50 = 26070 nM T28887 COV42L 137639829 IC50 > 30000 nM T28887 CL02GC 137640047 IC50 > 30000 nM T28887 CGKA54 137640295 IC50 > 30000 nM T28887 C7VIL6 137640304 IC50 > 30000 nM T28887 C0Q3ZW 137640468 IC50 > 30000 nM T28887 C7HF0W 137640828 IC50 = 181 nM T28887 CFQ9M8 137640986 IC50 = 240 nM T28887 C39FQX 137641152 IC50 > 30000 nM T28887 CSA84O 137641263 IC50 = 21790 nM T28887 CI4PM3 137641395 IC50 > 30000 nM T28887 C4OEC3 137641520 IC50 = 430 nM T28887 CS1K3I 137641616 IC50 > 30000 nM T28887 C38HXT 137641735 IC50 > 30000 nM T28887 CQ20LZ 137641789 IC50 = 286 nM T28887 CV19SL 137642038 IC50 > 30000 nM T28887 C6N0YZ 137642406 IC50 = 1020 nM T28887 C40JZA 137642448 IC50 > 30000 nM T28887 CY02GK 137642671 IC50 > 30000 nM T28887 C1PRH5 137642860 IC50 = 7330 nM T28887 CQF49N 137643043 IC50 = 35 nM T28887 C5QC2N 137643440 IC50 = 1220 nM T28887 C4V1WC 137643841 IC50 = 23480 nM T28887 CC38FN 137644424 IC50 > 30000 nM T28887 CVQ4J0 137644605 IC50 > 30000 nM T28887 CX37VS 137644658 IC50 > 30000 nM T28887 CPL3J1 137645258 IC50 > 30000 nM T28887 C8GNS5 137645287 IC50 = 16200 nM T28887 C8XAR3 137645372 IC50 > 30000 nM T28887 CI8YV3 137645454 IC50 = 151 nM T28887 C05LHW 137645511 IC50 > 30000 nM T28887 C2WO0K 137645865 IC50 = 4150 nM T28887 CYSU67 137645967 IC50 > 30000 nM T28887 CV7F6C 137646133 IC50 = 8110 nM T28887 CMJ7D9 137646202 IC50 > 30000 nM T28887 CN08DL 137646214 IC50 > 30000 nM T28887 CKL0A3 137646677 IC50 = 202 nM T28887 C4I9YE 137647260 IC50 = 8390 nM T28887 CX8C9V 137647325 IC50 > 30000 nM T28887 CA0V2Q 137647353 IC50 = 6760 nM T28887 CHW8X4 137647384 IC50 > 30000 nM T28887 CGMN16 137647616 Ki > 50000 nM T28887 CM65KH 137647813 IC50 > 100 nM T28887 CZ2RN9 137647935 IC50 > 30000 nM T28887 C8S2TO 137648573 IC50 > 30000 nM T28887 C0VAB8 137648585 IC50 > 30000 nM T28887 CPK7Y5 137648623 IC50 > 30000 nM T28887 CL0XW1 137648762 IC50 = 6720 nM T28887 CR0P6Z 137648837 IC50 = 29540 nM T28887 CG2PL8 137648996 IC50 > 30000 nM T28887 C05DNH 137649390 IC50 > 30000 nM T28887 CJA43U 137649535 IC50 = 136 nM T28887 CO20AE 137649565 IC50 > 30000 nM T28887 CGK2M9 137649620 IC50 = 9600 nM T28887 CDXE54 137649646 Ki > 50000 nM T28887 CH0ES8 137650022 IC50 > 30000 nM T28887 C15DRY 137650189 IC50 = 227 nM T28887 C4MC5X 137650991 IC50 > 30000 nM T28887 C3M0AW 137651229 IC50 = 120 nM T28887 C4GNA5 137651338 IC50 > 30000 nM T28887 CA0Z1V 137651534 IC50 = 335 nM T28887 CA4FM3 137651729 IC50 = 442 nM T28887 C8PWX1 137651771 IC50 > 30000 nM T28887 CGE1Z5 137651786 IC50 > 30000 nM T28887 CD89ZR 137651966 IC50 > 30000 nM T28887 CT05IE 137651994 IC50 > 30000 nM T28887 CH3B5G 137652131 IC50 > 30000 nM T28887 C5FHD3 137652442 IC50 = 200 nM T28887 CB15PI 137652670 Ki > 50000 nM T28887 C83RBI 137652888 IC50 = 8520 nM T28887 CSX6Q0 137652925 IC50 = 840 nM T28887 C7YS8U 137653259 IC50 = 175 nM T28887 C3XK2M 137653288 IC50 = 147 nM T28887 C61VOF 137653427 IC50 = 12670 nM T28887 CK4RS0 137653835 IC50 = 38 nM T28887 CXZ5J3 137654094 IC50 = 7400 nM T28887 C1OAE9 137654162 IC50 > 30000 nM T28887 CIW9C6 137654210 Ki = 999 nM T28887 C39QLZ 137654517 IC50 = 911 nM T28887 CFQ4T2 137654668 IC50 > 30000 nM T28887 CE75XW 137654719 IC50 = 130 nM T28887 CCR5B3 137654793 IC50 = 310 nM T28887 C1SBN5 137654946 IC50 = 390 nM T28887 CLWF87 137655165 IC50 > 30000 nM T28887 CS50BH 137655597 IC50 > 30000 nM T28887 CIA0V1 137656228 IC50 > 30000 nM T28887 CI6R3W 137656303 Ki > 50000 nM T28887 C76OGQ 137656942 IC50 = 1100 nM T28887 C5BM7T 137657586 IC50 > 100000 nM T28887 CR6B5H 137657803 IC50 = 69 nM T28887 C21XDS 137657845 IC50 = 380 nM T28887 C1DL3P 137657892 Ki > 50000 nM T28887 CA8J9V 137657988 IC50 = 2100 nM T28887 CN0C1E 137658519 IC50 > 30000 nM T28887 C8D2GT 137658785 Ki > 50000 nM T28887 COC9D2 137658833 IC50 > 30000 nM T28887 C3Q7PX 137660404 IC50 > 30000 nM T28887 C2RNY3 137661648 IC50 = 2530 nM T28887 CO7Q1H 137661848 IC50 = 248 nM T28887 CEJI95 137661885 IC50 = 3500 nM T28887 CI02VN 137662006 IC50 = 161 nM T28887 CQAY45 137662133 IC50 > 30000 nM T28887 CAQ62X 137701235 Ki = 110 nM T28887 CXV84M 138377596 IC50 = 2470 nM T28887 CVA12U 138377601 IC50 = 309 nM T28887 C7EM3I 138393071 IC50 = 646 nM T28887 C4NFS3 138393072 IC50 = 1224 nM T28887 CA3C4O 138454792 IC50 = 18 nM T28887 CN2UH1 139303146 IC50 = 16.84 nM T28887 C13JZX 141522811 IC50 = 80 nM T28887 CHS9N0 141728829 IC50 = 120 nM T28887 C9H8PX 141728841 IC50 = 840 nM T28887 CBV2K5 141728842 IC50 = 4070 nM T28887 C2HF9A 141728845 IC50 = 1700 nM T28887 C4RGY1 141728867 IC50 = 5100 nM T28887 CH9K7L 141733188 IC50 = 1480 nM T28887 C7XI0V 141764754 IC50 = 260 nM T28887 CX0E9B 142505968 IC50 = 353 nM T28887 C9G5ZW 142505990 IC50 = 3840 nM T28887 CBJC50 142505992 IC50 = 1937 nM T28887 CJ5GT3 142506013 IC50 = 71 nM T28887 C7N8LV 142506025 IC50 = 1758 nM T28887 CKBF56 142506033 IC50 = 385 nM T28887 CLND62 142506170 IC50 = 6194 nM T28887 CGNQ74 142506189 IC50 = 250 nM T28887 C1T3IQ 142506210 IC50 = 253 nM T28887 CEGV67 142506220 IC50 = 138 nM T28887 CP5HF8 142506225 IC50 = 320 nM T28887 C1COW3 145948735 IC50 = 1180 nM T28887 CZ6D7U 145948737 IC50 = 2230 nM T28887 CL1T5W 145948741 IC50 = 2530 nM T28887 C1GMF5 145948743 IC50 = 1840 nM T28887 CCEB28 145948752 IC50 = 877 nM T28887 CTO5X4 145948791 IC50 = 3200 nM T28887 CP98HY 145948798 IC50 > 10000 nM T28887 C43XJI 145948810 IC50 = 2770 nM T28887 C3JMP9 145948813 IC50 = 986 nM T28887 C7K1WB 145948814 IC50 = 2210 nM T28887 CFU6J8 145948816 IC50 = 7120 nM T28887 CG1Y3W 145948818 IC50 = 604 nM T28887 CAY43C 145948836 IC50 > 10000 nM T28887 CKI3Y2 145948841 IC50 = 314 nM T28887 C7JWF3 145948843 IC50 = 1440 nM T28887 CJG3B6 145948850 IC50 = 985 nM T28887 CGKI09 145948851 IC50 = 4300 nM T28887 CZ16SK 145948852 IC50 = 786 nM T28887 CA6W8I 145948853 IC50 = 2450 nM T28887 CF0Q3C 145948854 IC50 > 10000 nM T28887 CTEI37 145948871 IC50 = 1180 nM T28887 C0VTX8 145948874 IC50 > 10000 nM T28887 C8FHP2 145948903 IC50 = 5380 nM T28887 C7RLZ8 145948904 IC50 > 10000 nM T28887 CE4WS8 145948905 IC50 = 1700 nM T28887 C1KO6S 145948906 IC50 = 1820 nM T28887 C5EKH9 145948907 IC50 = 2370 nM T28887 C5HL4D 145948914 IC50 = 709 nM T28887 C74UFN 145948956 IC50 = 749 nM T28887 CY09KL 145948957 IC50 = 1090 nM T28887 CH91ER 145948958 IC50 > 10000 nM T28887 CE38KZ 145948959 IC50 = 644 nM T28887 CE15JW 145948961 IC50 = 1280 nM T28887 CN6YM2 145948964 IC50 = 10200 nM T28887 CY49SE 145948983 IC50 > 10000 nM T28887 CH0UZ1 145948985 IC50 = 4510 nM T28887 C7Y5PK 145948986 IC50 = 817 nM T28887 CY1KB9 145949010 IC50 = 713 nM T28887 CXJ0Y4 145949850 IC50 = 202 nM T28887 CRKM19 145950884 IC50 = 204 nM T28887 CV3QO5 145951170 IC50 = 752 nM T28887 CRSM78 145952088 IC50 = 75200 nM T28887 CKG98W 145953085 IC50 = 3050 nM T28887 CBNG29 145957781 IC50 = 295 nM T28887 C3L8IE 145958641 IC50 = 609 nM T28887 CO05IK 145959360 IC50 = 572 nM T28887 C9IV1C 145959866 IC50 = 560.9 nM T28887 CK1XI0 145960971 IC50 > 10000 nM T28887 C1X5EO 145962694 IC50 = 351 nM T28887 C29PAL 145963897 IC50 = 480 nM T28887 CJ47DY 145964043 IC50 = 6700 nM T28887 C3PWD4 145964064 IC50 = 2810 nM T28887 CEX67F 145964240 IC50 = 55 nM T28887 CDO47P 145964554 IC50 = 950 nM T28887 CDY56B 145964885 IC50 = 812 nM T28887 CB51JU 145965019 IC50 = 19000 nM T28887 CW6UM7 145965159 IC50 = 1800 nM T28887 C9XLE7 145966296 IC50 = 24200 nM T28887 CM6KY1 145966543 IC50 = 340 nM T28887 CJAE67 145966594 IC50 = 1490 nM T28887 CTUF34 145966712 IC50 = 1660 nM T28887 CTRI57 145966861 IC50 = 910 nM T28887 CUD38A 145967089 IC50 = 44 nM T28887 C19POY 145967140 IC50 = 1120 nM T28887 C93JKN 145967593 IC50 > 5000 nM T28887 CD82XB 145967610 IC50 > 5000 nM T28887 C7OG1D 145967698 IC50 > 5000 nM T28887 C5RPQ9 145967832 IC50 > 5000 nM T28887 CI1ZD2 145967851 IC50 > 5000 nM T28887 CR59HK 145967905 IC50 > 5000 nM T28887 C95SNQ 145967968 IC50 > 5000 nM T28887 CX0OD9 145968046 IC50 = 132.3 nM T28887 CES7W6 145968087 IC50 > 5000 nM T28887 CSO4I7 145968364 IC50 > 5000 nM T28887 C2XS8E 145968675 IC50 = 5500 nM T28887 CSJ81Y 145968726 IC50 = 2750 nM T28887 CG0S9U 145968824 IC50 > 5000 nM T28887 CIA79M 145968985 IC50 > 5000 nM T28887 C27YHM 145969456 IC50 = 2951 nM T28887 CV53YN 145969651 IC50 > 5000 nM T28887 C0K6XS 145969789 IC50 > 5000 nM T28887 CUI37A 145969799 IC50 = 354.2 nM T28887 CZ80EP 145969996 IC50 > 5000 nM T28887 C79YOL 145970069 IC50 = 82 nM T28887 CFL68X 145970091 IC50 = 33900 nM T28887 C7TSV2 145970161 IC50 > 5000 nM T28887 CG5OK8 145970171 IC50 = 3710 nM T28887 C3FQ0V 145970292 IC50 = 60 nM T28887 C8FXH4 145970309 IC50 = 210 nM T28887 CBR60K 145970453 IC50 > 5000 nM T28887 C0E2UO 145970598 IC50 > 5000 nM T28887 CI43DY 145970786 IC50 = 1260 nM T28887 C7K1AJ 145971681 IC50 = 6065 nM T28887 CW0T7A 145973234 IC50 = 2170 nM T28887 C4HTO2 145973543 IC50 = 1420 nM T28887 CSR50O 145973656 IC50 = 3000 nM T28887 CFP2R3 145973876 IC50 = 190 nM T28887 CVM0Z3 145974125 IC50 = 10000 nM T28887 CLCU89 145974270 IC50 = 1900 nM T28887 C8YEJ9 145974425 IC50 = 1240 nM T28887 C5YJO8 145974667 IC50 = 10000 nM T28887 CZL05M 145975187 IC50 = 3500 nM T28887 CE8I5V 145975869 IC50 = 3530 nM T28887 C6Y9QH 145975913 IC50 = 110 nM T28887 CU65BZ 145976000 IC50 = 9200 nM T28887 C7ANI4 145976192 IC50 = 380 nM T28887 C86GXV 145976671 IC50 = 390 nM T28887 CMUA94 145976675 IC50 = 4480 nM T28887 CN6UO4 145977003 IC50 = 5340 nM T28887 CKAQ67 145977127 IC50 = 756 nM T28887 C78XNS 145977336 IC50 = 19000 nM T28887 CP53JS 145977717 IC50 = 398.3 nM T28887 C3QYB8 145978561 IC50 = 19000 nM T28887 COR40V 145978805 IC50 = 1060 nM T28887 CZ7IQ9 145979841 IC50 = 875 nM T28887 CMB08D 145981960 IC50 > 30000 nM T28887 C9VDE5 145982499 IC50 = 1550 nM T28887 C6OL1K 145983267 IC50 = 1960 nM T28887 CWD0A9 145983712 Ki = 100 nM T28887 C17UTC 145983813 IC50 = 1550 nM T28887 CIWO70 145984314 IC50 = 1220 nM T28887 C9ZKC1 145984665 IC50 = 1670 nM T28887 CN6KB9 145985243 IC50 = 284 nM T28887 C56MWZ 145986208 Ki = 320 nM T28887 CL62QV 145986214 IC50 = 2940 nM T28887 C51BUM 145986322 IC50 > 1000 nM T28887 C1WH7V 145986586 IC50 > 5000 nM T28887 C7L1GU 145986811 IC50 = 47.3 nM T28887 CFWH51 145987165 IC50 = 1602 nM T28887 CRX8H1 145987492 IC50 > 5000 nM T28887 CPAX89 145987732 IC50 > 5000 nM T28887 CJ1M7T 145987832 IC50 = 1115 nM T28887 C82CIN 145988785 IC50 > 30000 nM T28887 CJ8DO3 145989487 IC50 > 5000 nM T28887 CO4J2D 145990209 EC50 = 341000 nM T28887 CHR0U9 145990400 IC50 > 1000 nM T28887 C4PSZ2 145990543 IC50 = 253 nM T28887 CF54BR 145993638 IC50 = 1344 nM T28887 C1W6CF 145994016 IC50 = 290 nM T28887 C0GMR1 146585718 IC50 = 204 nM T28887 C0YXS8 147254231 IC50 = 599 nM T28887 C48EXH 148289288 IC50 = 165.5 nM T28887 C3SA6B 148608442 IC50 = 4910 nM T28887 CO47EC 148970856 IC50 = 3880 nM T28887 CN71OS 149405396 IC50 > 100000 nM T28887 CV5ZR0 149819902 IC50 = 1640 nM T28887 CH3JE4 150054712 IC50 = 1049 nM T28887 C8S3MF 150076000 IC50 > 300 nM T28887 CU2XY0 150312795 IC50 = 3060 nM T28887 C5PQI9 150470306 IC50 = 1068 nM T28887 C4JP7X 150533939 IC50 = 2751 nM T28887 CAQ36F 150619353 IC50 = 1760 nM T28887 C89BKD 150622000 IC50 = 653 nM T28887 CIM06Z 150916115 IC50 = 1442 nM T28887 CM6IF7 151532669 IC50 = 845 nM T28887 CS0V6U 151543423 IC50 = 1155 nM T28887 CV39LB 151825687 IC50 = 1191 nM T28887 CA21YZ 151887635 IC50 = 731 nM T28887 CROU95 152148008 IC50 = 169 nM T28887 CY1NG0 152157103 IC50 = 2521 nM T28887 CYF2I5 152375216 IC50 = 97 nM T28887 CL1UA7 152547478 IC50 = 95 nM T28887 C2AOQ6 152562172 IC50 = 429 nM T28887 CT4H9P 153408403 IC50 = 525 nM T28887 CK7P3F 153408410 IC50 = 1150 nM T28887 C9FIY4 153534005 IC50 = 167 nM T28887 C7F1UK 155454897 IC50 = 2000 nM T28887 CQ5BL7 155512551 IC50 = 1000 nM T28887 CPF6R7 155512997 IC50 = 133 nM T28887 C7VKU2 155513116 IC50 > 32000 nM T28887 CE4H7I 155513471 IC50 = 13000 nM T28887 CW3VT9 155514603 IC50 = 1600 nM T28887 CH4UZ2 155514990 IC50 = 8 nM T28887 CZ84WI 155515284 IC50 = 600 nM T28887 CWEZ05 155515488 IC50 = 0.41 nM T28887 CUKG21 155515602 IC50 = 1200 nM T28887 CY2DC1 155515836 IC50 > 1000 nM T28887 CYJ53T 155515864 IC50 = 76 nM T28887 CA1J3N 155517086 IC50 = 6700 nM T28887 CL72ME 155517175 IC50 = 1755 nM T28887 CY54TU 155518062 IC50 = 1900 nM T28887 CEH2N5 155518106 IC50 > 100000 nM T28887 C58ZNC 155518327 IC50 = 27.14 nM T28887 CCDU61 155518496 IC50 > 32000 nM T28887 C41AIO 155518963 IC50 > 1000 nM T28887 CAD06U 155519254 IC50 = 920 nM T28887 CDY5H6 155519645 IC50 = 3410 nM T28887 CAZ3S7 155521187 IC50 = 2000 nM T28887 CZ75FW 155521272 IC50 = 3600 nM T28887 CG4F2U 155521283 IC50 > 32000 nM T28887 C0YB4H 155521454 IC50 = 2300 nM T28887 CEQ58R 155523224 IC50 > 1000 nM T28887 CU5RZ1 155524034 IC50 = 400 nM T28887 CNW0D1 155524821 IC50 = 617 nM T28887 CN7B1T 155525782 IC50 > 100000 nM T28887 C71UNO 155527385 Ki = 4700 nM T28887 CHR4K5 155528532 IC50 > 100000 nM T28887 CQ4RG3 155528629 IC50 = 4070 nM T28887 C0IC6W 155528706 IC50 > 1000 nM T28887 CZ70PO 155529066 IC50 = 31000 nM T28887 C49NGT 155529137 IC50 = 1000 nM T28887 C9L6OC 155529247 IC50 = 12 nM T28887 CZMC49 155530597 IC50 = 787 nM T28887 COTR30 155530602 IC50 = 573 nM T28887 C47WTL 155531016 IC50 = 620 nM T28887 CN3W5J 155531452 IC50 = 5400 nM T28887 CK2UY4 155531957 IC50 = 370 nM T28887 C3HDI1 155532640 IC50 = 44.09 nM T28887 CD8ZV7 155532950 IC50 = 29900 nM T28887 CIZ46A 155533876 IC50 = 2900 nM T28887 CPE68B 155534222 IC50 = 794.33 nM T28887 C6LB5D 155535084 IC50 = 5300 nM T28887 CK8SD7 155535151 IC50 = 9100 nM T28887 CJH9L4 155535498 IC50 > 1000 nM T28887 C2JH0S 155537112 IC50 = 9210 nM T28887 CTF98X 155537473 IC50 = 1520 nM T28887 CAG9P4 155537573 IC50 = 260 nM T28887 CCD7Z8 155538128 IC50 = 4 nM T28887 C63FKN 155538445 IC50 > 10000 nM T28887 C1PFV7 155538765 IC50 = 255 nM T28887 CLD19W 155539311 IC50 = 422 nM T28887 CU6V4Q 155539319 IC50 = 12000 nM T28887 C6U0FM 155540189 IC50 = 130 nM T28887 CKZ9A5 155543845 IC50 = 85.4 nM T28887 C4DQ8E 155544048 IC50 = 133 nM T28887 CP4L1F 155544459 IC50 = 420 nM T28887 CJK31W 155544599 IC50 = 4090 nM T28887 C1VF5A 155544728 IC50 = 224 nM T28887 CTN47R 155544947 IC50 = 3 nM T28887 CXR86J 155545078 IC50 = 7800 nM T28887 CCV9J0 155545380 IC50 = 8.5 nM T28887 CWS48H 155545802 IC50 = 160 nM T28887 C7YOP9 155545823 IC50 = 1700 nM T28887 CF2O4J 155546325 IC50 = 2300 nM T28887 CK45LA 155546486 IC50 = 794.33 nM T28887 C3HB0U 155546555 IC50 = 398.11 nM T28887 CS3GO2 155546558 IC50 = 2460 nM T28887 C0AU1L 155546632 IC50 = 1000 nM T28887 CEF69A 155546817 IC50 > 1000 nM T28887 CHD0I6 155547367 IC50 = 719 nM T28887 C1D4PI 155547606 Ki = 4210 nM T28887 C90FBZ 155549087 IC50 > 50000 nM T28887 CCTU12 155549163 IC50 > 1000 nM T28887 CE0YL6 155549538 IC50 > 30000 nM T28887 CO6ID4 155550122 IC50 = 14100 nM T28887 C4Z5JX 155550827 IC50 = 7000 nM T28887 CU74MG 155550898 IC50 = 7 nM T28887 CA03BO 155551057 IC50 = 398.11 nM T28887 CEO4J8 155551917 IC50 = 423.1 nM T28887 C05ZVG 155552130 IC50 = 819 nM T28887 C46WHP 155552329 IC50 > 1000 nM T28887 CCUO56 155552443 IC50 = 19700 nM T28887 CV4Y5B 155552792 IC50 > 30000 nM T28887 CGDF76 155554360 IC50 = 1100 nM T28887 CC56ED 155554844 IC50 = 2580 nM T28887 C3OEL8 155554927 IC50 = 1500 nM T28887 CXGR50 155555191 IC50 > 30000 nM T28887 CFW90N 155555562 IC50 = 35.67 nM T28887 C7QTU1 155555957 IC50 = 30000 nM T28887 CIN57Q 155556138 IC50 = 1260 nM T28887 C0IO1Q 155557341 IC50 > 1000 nM T28887 CJ9FW6 155557777 IC50 = 635 nM T28887 CJ3MZ1 155558467 IC50 = 28 nM T28887 C8AUB0 155558567 IC50 = 1080 nM T28887 C0RZ7V 155558710 IC50 > 1000 nM T28887 C2IS1E 155559200 IC50 = 229.2 nM T28887 C28CVZ 155559279 IC50 = 90.6 nM T28887 CPD50Q 155559583 IC50 = 1600 nM T28887 CY3XI1 155559600 IC50 > 1000 nM T28887 CC62UI 155559872 IC50 > 10000 nM T28887 CMD6Q7 155560250 IC50 = 1400 nM T28887 CGL24S 155562249 IC50 = 170 nM T28887 C9UYZ6 155564157 IC50 = 243.1 nM T28887 C4IM1X 155564305 IC50 = 37.9 nM T28887 CX23YB 155564400 IC50 = 378 nM T28887 CPNA06 155564750 IC50 = 1300 nM T28887 C87JXN 155564870 IC50 = 316.23 nM T28887 CE0U7K 155564881 IC50 > 1000 nM T28887 CZDC03 155565491 IC50 = 6700 nM T28887 CG65CR 155565674 IC50 = 1200 nM T28887 C3G1JV 155565712 IC50 > 1000 nM T28887 CD05RS 155566122 IC50 = 2300 nM T28887 C4A0RK 155566461 IC50 = 13000 nM T28887 C51BFK 155566644 IC50 = 3130 nM T28887 C04CGS 155567444 IC50 = 1600 nM T28887 CT6Z4H 155567814 IC50 = 65.7 nM T28887 CS03PJ 155568350 IC50 = 1700 nM T28887 C1S7AP 155568542 IC50 = 464 nM T28887 C5NQK8 155569352 IC50 = 281.1 nM T28887 CW5XB4 155569484 IC50 > 30000 nM T28887 D00DQZ 11964504 IC50 = 190 nM T28887 D00GBB 11449246 Ki = 252 nM T28887 D00KFF 9882812 Ki = 33 nM T28887 D00SEE 11379392 IC50 = 1070 nM T28887 D01BCK 23382 IC50 = 14000 nM T28887 D01FYB 23648267 IC50 > 20000 nM T28887 D01YBR 44591988 IC50 = 235 nM T28887 D02NWS 279980 Ki = 1850 nM T28887 D03HNC 17748273 IC50 = 300 nM T28887 D03QOD 239512 IC50 = 43000 nM T28887 D03ZUZ 11381650 IC50 = 405 nM T28887 D04KQF 6675804 Ki = 143.1 nM T28887 D04UVL 1133083 IC50 > 50000 nM T28887 D05OVV 11993691 IC50 = 240 nM T28887 D05QBX 44369352 IC50 = 20000 nM T28887 D06THS 25151110 IC50 = 2320 nM T28887 D07MYE 5355635 IC50 = 759 nM T28887 D07YZZ 5173 Ki = 950 nM T28887 D09LVY 11964503 IC50 = 690 nM T28887 D09RKA 72946782 IC50 = 5000 nM T28887 D0B3ZM 11436024 IC50 = 1360 nM T28887 D0D7KH 25151675 IC50 = 7130 nM T28887 D0E0TA 44454650 IC50 > 50000 nM T28887 D0E9DD 16095101 IC50 = 3700 nM T28887 D0G6DH 16661454 IC50 = 690 nM T28887 D0H3RO 25190758 IC50 = 11050 nM T28887 D0H4YW 3611 Ki = 177.95 nM T28887 D0I5XM 25152062 IC50 = 4730 nM T28887 D0K7QR 45269423 IC50 = 600 nM T28887 D0L7HP 6675803 Ki = 750 nM T28887 D0M9LJ 44454415 IC50 > 50000 nM T28887 D0MD7H 44454143 IC50 > 50000 nM T28887 D0N9AK 44138031 IC50 = 1290 nM T28887 D0O7UF 10923922 IC50 = 450 nM T28887 D0P3SU 10192705 IC50 = 6600 nM T28887 D0P9CQ 25151109 IC50 = 6680 nM T28887 D0Q2GM 44454416 IC50 > 50000 nM T28887 D0Q5DI 71462653 IC50 = 1540 nM T28887 D0Q5MC 24753719 IC50 = 6.6 nM T28887 D0Q9PO 16095114 Ki > 5000 nM T28887 D0QX6R 10998964 IC50 = 1500 nM T28887 D0R2HF 11437457 IC50 = 3890 nM T28887 D0R7JA 53344908 Ki = 2706 nM T28887 D0S0WK 11075845 IC50 = 500 nM T28887 D0T0BE 11426781 IC50 = 270 nM T28887 D0T0SK 44138032 IC50 = 70 nM T28887 D0T4JQ 264 IC50 = 15000 nM T28887 D0U8FC 759408 IC50 > 50000 nM T28887 D0V1HA 24880249 IC50 = 700 nM T28887 D0W1PV 6918328 Ki = 49 nM T28887 D0X4VO 44359538 IC50 = 22000 nM T28887 D0XZ9Q 11149404 IC50 = 1120 nM T28887 D0YO6M 785232 IC50 > 20000 nM T28887 D0Z2VP 11139963 IC50 = 65 nM T28887 D0Z8PX 24757913 IC50 = 120 nM T15776 D0EG1I 9926791 IC50 > 10000 nM T15776 D01FQV 517326 EC50 = 5700000 nM T15776 D03HUX 49792852 IC50 > 10000 nM T15776 D03LWG 53235510 IC50 > 10000 nM T15776 D05PZB 135398495 IC50 = 10 nM T15776 D07DTV 11338033 IC50 > 10000 nM T15776 D0E3TC 44259 IC50 = 0.506 nM T15776 D0P1CV 46191454 IC50 > 10000 nM T15776 D0Z1DH 10029385 IC50 = 6200 nM T15776 D03BNU 59604787 IC50 > 3500 nM T15776 D03GFC 16741245 IC50 = 41 nM T15776 D0T3ME 156422 IC50 > 30000 nM T15776 CHGI09 6597 IC50 = 1025000 nM T15776 CM75BH 8447 IC50 = 379 nM T15776 CMC1D0 12892 IC50 = 49 nM T15776 C2NY3B 357976 IC50 = 326 nM T15776 C07TEG 764764 IC50 = 648000 nM T15776 C6NQ9Y 1116656 IC50 = 290 nM T15776 C1TX7F 3467157 IC50 = 161 nM T15776 CDK3J0 5703619 IC50 = 8.3 nM T15776 CNP39D 6102761 IC50 = 66 nM T15776 CG7X9S 7178546 EC50 = 11700 nM T15776 CN6FO5 9850141 IC50 = 300 nM T15776 C7SFI1 10296883 IC50 = 6700 nM T15776 C7HBP6 10429593 IC50 > 10000 nM T15776 C30PKR 11248978 IC50 > 20000 nM T15776 CSXY78 11294864 IC50 = 4300 nM T15776 CPU9I3 11316975 IC50 > 20000 nM T15776 CQ8I4H 11328863 IC50 = 6500 nM T15776 C43NPS 11373886 IC50 > 10000 nM T15776 C0H6QS 11495680 IC50 > 10000 nM T15776 CIW9L5 11502867 IC50 > 10000 nM T15776 CK2Q0X 11516978 IC50 > 10000 nM T15776 CPE53F 11526238 IC50 > 10000 nM T15776 C7HMO6 11526786 IC50 > 200000 nM T15776 C5BM4T 11531799 IC50 > 10000 nM T15776 C53OSD 11532048 IC50 > 10000 nM T15776 CC4QM5 11532676 IC50 > 10000 nM T15776 CTG83F 11539329 Ki > 3800 nM T15776 C01FVM 11546457 IC50 > 10000 nM T15776 CNBM81 11562171 IC50 > 10000 nM T15776 CO9KP5 11583459 IC50 > 30000 nM T15776 CMIL86 11590363 Ki > 3800 nM T15776 C0NV9Y 11596881 IC50 > 10000 nM T15776 C1BLZ5 11620055 IC50 > 10000 nM T15776 C9T6SC 11640926 Ki > 3800 nM T15776 C24GRQ 11661959 IC50 > 10000 nM T15776 CS72ED 11682843 IC50 > 10000 nM T15776 CLC53E 11691173 IC50 > 10000 nM T15776 C1FTX3 11719305 IC50 > 10000 nM T15776 C9JT4S 11847343 IC50 = 762 nM T15776 CC28SV 16414363 IC50 = 3140 nM T15776 CHK6P1 16424570 IC50 = 2970 nM T15776 CEL0F3 20537765 IC50 = 109 nM T15776 CTF23G 20644743 IC50 > 50000 nM T15776 CZ7V8L 21048651 IC50 > 100000 nM T15776 CAJ4T2 24762205 IC50 > 10000 nM T15776 CJUK39 24770517 IC50 > 10000 nM T15776 C0EKO5 24772654 IC50 > 10000 nM T15776 C9PA0M 24807809 IC50 > 200000 nM T15776 C13QYB 24884503 IC50 > 2000 nM T15776 C6CVK4 24959046 IC50 > 100000 nM T15776 CD5HQ0 24969301 IC50 > 10000 nM T15776 C4EG8R 24993189 IC50 > 10000 nM T15776 CNG96H 25210579 IC50 > 10000 nM T15776 CRO09K 25211064 IC50 = 3100 nM T15776 C75HIL 28099854 EC50 = 4640 nM T15776 CKQY13 28361735 IC50 = 5900 nM T15776 C28NIL 29255080 IC50 = 410 nM T15776 C0RCX1 42196244 EC50 = 500 nM T15776 CO4PL8 42606076 IC50 = 12600 nM T15776 C20VGT 42606077 IC50 = 3870 nM T15776 C7N5EC 42606078 IC50 = 39200 nM T15776 CI69YO 42606079 IC50 > 100000 nM T15776 C5L7IT 42606080 IC50 = 20800 nM T15776 CG04LZ 42606083 IC50 > 100000 nM T15776 C0WEU1 42606190 IC50 > 100000 nM T15776 CD6LN3 42606191 IC50 > 25000 nM T15776 CWR7P5 42606194 IC50 > 100000 nM T15776 CJ2GM1 42606195 IC50 > 100000 nM T15776 C61JUL 42606196 IC50 > 100000 nM T15776 C9GS8P 42606431 IC50 > 50000 nM T15776 CV09DY 44410717 IC50 > 10000 nM T15776 CP3CI1 44410720 IC50 > 10000 nM T15776 C8W7AD 44410723 IC50 > 10000 nM T15776 CAT5X4 44410829 IC50 > 10000 nM T15776 CC6Y5P 44410844 IC50 > 10000 nM T15776 CG34TY 44410851 IC50 > 10000 nM T15776 C41EIA 44410869 IC50 > 10000 nM T15776 CB6AE8 44410948 IC50 > 10000 nM T15776 CXZG12 44410949 IC50 > 10000 nM T15776 CS7IE9 44410953 IC50 > 10000 nM T15776 CA9M4X 44410954 IC50 > 10000 nM T15776 C3SP5H 44410955 IC50 > 10000 nM T15776 C5D6YP 44410956 IC50 > 10000 nM T15776 C5W1VC 44410959 IC50 > 10000 nM T15776 CM1C2G 44410960 IC50 > 10000 nM T15776 CVSI80 44411048 IC50 > 10000 nM T15776 CN72BR 44411161 IC50 > 10000 nM T15776 C4AW0O 44411183 IC50 > 10000 nM T15776 C5Z3LI 44591740 IC50 > 30000 nM T15776 CU3RF1 45139989 IC50 > 10000 nM T15776 CQGZ06 45139991 IC50 > 10000 nM T15776 C7ON5A 46233287 IC50 > 10000 nM T15776 C7H4YM 46865419 IC50 > 10000 nM T15776 CQR9K1 46933384 IC50 > 100000 nM T15776 C2B5XF 49765254 IC50 > 10000 nM T15776 CJZ5A0 49840306 IC50 > 10000 nM T15776 CA4NH7 49850583 IC50 > 50000 nM T15776 CT4Y6E 49852123 IC50 > 100000 nM T15776 C83VHI 49864785 IC50 > 100000 nM T15776 C2UTK6 49864850 IC50 > 100000 nM T15776 CAE53W 49865153 IC50 > 100000 nM T15776 C2W9OA 53324451 IC50 > 10000 nM T15776 C8NA4L 53384644 IC50 > 30000 nM T15776 CE1ZK6 54759168 IC50 > 10000 nM T15776 C1XS2J 54760383 IC50 > 10000 nM T15776 CN9QD7 56643097 IC50 > 10000 nM T15776 CBOD63 56835089 IC50 > 30000 nM T15776 CD6Y9Z 57395116 IC50 > 30000 nM T15776 C8W6IG 57395117 IC50 > 30000 nM T15776 CG7S0D 57396882 IC50 > 30000 nM T15776 C80ODY 67932020 Ki = 1930 nM T15776 C5DGR9 69036886 IC50 = 136 nM T15776 CH0B8N 70789756 IC50 > 30000 nM T15776 CCN01X 71547862 IC50 > 10000 nM T15776 CA3O6K 71552696 IC50 > 30000 nM T15776 C1NPL0 71552941 IC50 > 30000 nM T15776 CA4PS8 71552942 IC50 > 30000 nM T15776 CELO13 72376512 IC50 = 2100 nM T15776 C47XUW 86280454 Ki = 28 nM T15776 COG97V 86346643 IC50 = 420 nM T15776 CY0UC4 90645194 IC50 > 10000 nM T15776 C19SVO 91827516 IC50 = 710 nM T15776 CI7HO1 97281116 IC50 = 1260 nM T15776 CC74KU 97444773 EC50 = 420 nM T15776 CK15CW 117967655 Ki = 200 nM T15776 CJ5F0T 117967696 Ki = 1170 nM T15776 CQ4FL0 117968039 Ki = 90 nM T15776 CYG8C4 117970892 Ki = 37 nM T15776 CZ2AI8 117972517 Ki = 26 nM T15776 CFI2P0 117972524 Ki = 67 nM T15776 CML61N 117972616 Ki = 980 nM T15776 C5TFJ0 117972658 Ki = 37 nM T15776 CK6QG0 117972799 IC50 = 109 nM T15776 CL57JX 122186227 IC50 = 56 nM T15776 CQ82GU 124201644 Ki = 124 nM T15776 C3FC0O 126200721 IC50 = 890 nM T15776 CBXH95 127024111 IC50 = 135 nM T15776 CS1ZO6 127024161 Ki = 16 nM T15776 CHQ12D 127024491 Ki = 241 nM T15776 CBS1R8 127024554 IC50 = 198 nM T15776 CR6A9C 127024644 IC50 = 15 nM T15776 CKQ63N 134561155 IC50 = 2060 nM T15776 CDU8E6 135517488 IC50 = 11900 nM T15776 CTJ48K 135524085 IC50 = 3300 nM T15776 CUT1W7 135524168 IC50 = 2200 nM T15776 CEK31P 135566415 IC50 > 20000 nM T15776 CX4ZB3 135863110 IC50 = 17000 nM T15776 CHA4N2 136013680 IC50 > 10 nM T15776 CX08NH 136087015 IC50 = 2949 nM T15776 C41VCO 136087016 IC50 = 1417 nM T15776 CSP52I 136087017 IC50 = 521 nM T15776 CG86UM 136087018 IC50 = 878 nM T15776 C6HBO1 136087019 IC50 = 776 nM T15776 CL4JQ2 136087020 IC50 = 952 nM T15776 C8W3YG 136087021 IC50 = 604 nM T15776 C2Y9KG 136087022 IC50 = 2369 nM T15776 CMD24T 136087023 IC50 = 4306 nM T15776 CYN98E 136087024 IC50 = 1070 nM T15776 C1BNT0 136087025 IC50 = 1050 nM T15776 C1DCG4 136087026 IC50 = 491 nM T15776 C7OM6G 136087027 IC50 = 557 nM T15776 CFN04C 136087028 IC50 = 845 nM T15776 CYN8W9 136087029 IC50 = 1916 nM T15776 C2DHJ6 136087030 IC50 = 28 nM T15776 CW4RY9 136087031 IC50 = 68 nM T15776 C6KI1S 136087032 IC50 = 17 nM T15776 C58XIU 136087033 IC50 = 160 nM T15776 CS6DX7 136087034 IC50 = 59 nM T15776 CQ64WB 136087035 IC50 = 150 nM T15776 CUCJ68 136087036 IC50 = 130 nM T15776 CKE0D9 136087037 IC50 = 210 nM T15776 CQ0HB5 136087038 IC50 > 10000 nM T15776 CI3WQ4 136087039 IC50 = 25 nM T15776 C0XOB5 136087040 IC50 = 580 nM T15776 CW87ZT 136087041 IC50 = 380 nM T15776 C2YIH8 136087042 IC50 = 610 nM T15776 C8N1QK 136167232 Ki = 136 nM T15776 C1YUD0 136219394 IC50 > 10 nM T15776 CH92BK 136249157 EC50 = 1990 nM T15776 C0BUJ9 136249185 IC50 = 620 nM T15776 CIU8W3 136254389 IC50 > 10 nM T15776 CV6KR8 137349062 IC50 = 67000 nM T15776 C7YW9Z 137632776 IC50 = 101 nM T15776 C0MC8O 137633010 IC50 = 130 nM T15776 C8C3NP 137633259 IC50 = 32 nM T15776 CV96IR 137634660 IC50 = 139 nM T15776 CZB16R 137636312 IC50 = 2437 nM T15776 CW3PS2 137636424 IC50 = 1701 nM T15776 C7PN8I 137636522 IC50 = 2854 nM T15776 CGT0C3 137637525 IC50 = 609 nM T15776 CW9GK1 137638442 IC50 > 10000 nM T15776 CIVP30 137639033 IC50 = 1048 nM T15776 CC7D8X 137641144 IC50 = 3875 nM T15776 CDC7X9 137642124 IC50 = 96 nM T15776 CFZX56 137644518 IC50 = 39 nM T15776 C6MLR7 137644803 IC50 = 119 nM T15776 CRSX58 137645173 IC50 = 588 nM T15776 CSD3C1 137645391 IC50 = 247 nM T15776 C69THL 137645576 IC50 > 10000 nM T15776 COD3J2 137645748 IC50 = 395 nM T15776 CV0FZ1 137647811 IC50 = 90 nM T15776 C2T6QV 137648710 IC50 = 90 nM T15776 CF7IU4 137648813 IC50 = 30 nM T15776 CDP6H0 137649627 IC50 = 6832 nM T15776 C65NKC 137650100 IC50 = 85 nM T15776 C5L1FM 137650751 IC50 = 169 nM T15776 C9K6EZ 137652154 IC50 = 702 nM T15776 CI5TH3 137653481 IC50 = 24 nM T15776 C43WDJ 137655420 IC50 = 109 nM T15776 C3PLK1 137655575 IC50 = 350 nM T15776 CES39P 137657445 IC50 = 113 nM T15776 C3DXH1 137658288 IC50 = 218 nM T15776 C3R4ZW 137659397 IC50 = 72 nM T15776 C3SV7G 137659540 IC50 = 26 nM T15776 C38XIS 137660188 IC50 = 289 nM T15776 CO6XK1 137660391 Ki = 260 nM T15776 CIR0N7 137660550 IC50 = 622 nM T15776 CO3Z2S 137660588 IC50 = 126 nM T15776 CA2CB9 137661423 IC50 = 1459 nM T15776 C49ZBX 137661735 IC50 = 476 nM T15776 C49JZI 137661912 IC50 = 2414 nM T15776 CL6T4P 149986651 IC50 = 36 nM T15776 C24DWX 150179460 IC50 = 151 nM T15776 CJ17UR 150426809 IC50 = 42 nM T15776 C1Z5DA 151004457 IC50 = 14 nM T15776 C02NBO 151026196 IC50 = 48 nM T15776 C0Q9PK 151406722 IC50 = 24 nM T15776 C2RVC3 151777753 IC50 = 20 nM T15776 CKR2T1 151835909 IC50 = 67 nM T15776 CTI5R1 151961601 IC50 = 113 nM T15776 CC3ME1 152131905 IC50 = 9 nM T15776 CAR6N3 152143591 IC50 = 24 nM T15776 C79SKI 152618834 IC50 = 140 nM T15776 CCG7K6 155528322 IC50 = 20 nM T15776 C8EH6M 155538895 IC50 = 57 nM T15776 D00ERW 44444843 Ki = 3482 nM T15776 D00HVA 11624601 Ki > 3800 nM T15776 D03DZO 11715767 IC50 > 10000 nM T15776 D06ZIO 44464263 IC50 = 421 nM T15776 D08HFG 24809764 IC50 > 10000 nM T15776 D09HVH 135566652 IC50 > 10 nM T15776 D0D9PD 11656591 IC50 > 5000 nM T15776 D0J3LR 11634725 Ki > 10000 nM T15776 D0L2WP 46225540 IC50 = 50 nM T15776 D0Q3NG 11715520 Ki > 3800 nM T15776 D0RG0Z 10077147 IC50 = 65 nM T15776 D0S7IE 11658882 Ki > 3800 nM T15776 D0T8NU 16757525 IC50 > 4000 nM T15776 D0Y5RO 4566 IC50 = 800 nM T15776 D0ZA6G 6323491 IC50 = 230000 nM T38338 D01NLB 16135415 IC50 = 500 nM T38338 D05CEU 941361 IC50 = 1670 nM T38338 D0N3ZJ 3949 IC50 = 2430 nM T38338 D05ADP 160355 EC50 = 27580 nM T38338 D0N3SR 5282138 IC50 = 1600 nM T38338 D0W8XT 60663 IC50 = 1340 nM T38338 D00BPA 4592 EC50 > 1000000 nM T38338 D03QMS 9956291 IC50 = 460 nM T38338 D0G6HZ 136180343 IC50 = 4400 nM T38338 D0IU2F 4988454 IC50 = 39000 nM T38338 CBF50H 244076 IC50 > 10000 nM T38338 C15GWK 512292 EC50 > 1000000 nM T38338 CE37GH 3579860 IC50 = 1680 nM T38338 CFK53N 3699946 IC50 = 660 nM T38338 CW2UD8 4099361 IC50 = 4800 nM T38338 CKP08L 5289296 EC50 > 1000000 nM T38338 CJ23HP 5494414 EC50 = 80000 nM T38338 C2XC5V 6603989 EC50 = 570000 nM T38338 CJ4U3H 6610355 EC50 > 1000000 nM T38338 C6CL7Q 9800610 IC50 = 210 nM T38338 CAX87O 9807599 IC50 = 290 nM T38338 C0WG2Y 9808556 IC50 = 340 nM T38338 CLX43S 9827369 IC50 = 1100 nM T38338 C18DRL 9849674 IC50 = 320 nM T38338 CQ4LC2 9872676 Ki = 5240 nM T38338 C0I1EJ 9873591 IC50 = 330 nM T38338 CP4AK0 9875854 IC50 = 490 nM T38338 C41XHA 9895079 IC50 = 200 nM T38338 CJUV43 9910160 IC50 = 4500 nM T38338 C5Z8XC 10004622 IC50 = 670 nM T38338 C0FYT4 10090396 IC50 = 10700 nM T38338 CTHX18 10090843 IC50 = 1330 nM T38338 CZG60Q 10137573 EC50 > 100000 nM T38338 CZN61C 10224083 IC50 = 630 nM T38338 C41AVB 10246646 IC50 = 880 nM T38338 C6U9MD 10247627 EC50 > 100000 nM T38338 CBU78F 10316864 IC50 = 1290 nM T38338 C8RJI5 10320344 IC50 = 500 nM T38338 CSRL36 10342500 IC50 = 700 nM T38338 C5ET8J 10348294 IC50 = 180 nM T38338 C6CGJ8 10362524 IC50 = 600 nM T38338 CJI2F0 10404129 IC50 = 490 nM T38338 C2BT1H 10404882 IC50 = 530 nM T38338 C8BFT9 10414472 IC50 = 2700 nM T38338 CZ9E7W 10425676 IC50 = 3980 nM T38338 C5LEY9 10427267 IC50 = 510 nM T38338 CZ9F3G 10431256 IC50 = 630 nM T38338 C5MXP3 10436852 IC50 = 3300 nM T38338 CTQ10K 10439014 IC50 = 740 nM T38338 CL35CW 10452361 IC50 = 1070 nM T38338 C8P7DV 10507403 IC50 = 260 nM T38338 CDM31B 10626133 IC50 = 480 nM T38338 C72TBJ 10626745 IC50 = 1000 nM T38338 CMK89L 10641624 IC50 = 4700 nM T38338 CD1FZ9 10696911 IC50 = 750 nM T38338 C56IES 10697309 IC50 = 2500 nM T38338 CZWI43 10697833 IC50 = 510 nM T38338 C2X6FH 10746013 IC50 = 4600 nM T38338 C2W6VR 10768986 IC50 = 830 nM T38338 CR7JE9 10841432 IC50 = 430 nM T38338 C4Q0HN 11202434 IC50 = 400 nM T38338 C7WJ0G 11349947 IC50 = 2400 nM T38338 CD3LV1 11398205 IC50 = 3100 nM T38338 CO9LU2 11541311 IC50 = 1700 nM T38338 CIVU58 11741229 IC50 = 1370 nM T38338 CA41XH 11742682 IC50 = 1320 nM T38338 C30UCP 11801527 IC50 = 1500 nM T38338 CEA98S 14774397 IC50 = 3500 nM T38338 C4KUX1 15487532 IC50 = 2800 nM T38338 C4BW7P 15487533 IC50 = 1900 nM T38338 CH3IX2 15487534 IC50 = 4100 nM T38338 C46WTA 15487535 IC50 = 1200 nM T38338 C04ERU 15487536 IC50 = 2600 nM T38338 CT8D4I 15487537 IC50 = 13000 nM T38338 C6W9GK 15487538 IC50 = 660 nM T38338 CCV1Q0 15487539 IC50 = 1100 nM T38338 COG71D 15487540 IC50 = 590 nM T38338 CXA3B9 15487541 IC50 = 880 nM T38338 CYF0I9 15487542 IC50 = 1200 nM T38338 CD7B8P 15487543 IC50 = 200 nM T38338 C1O2ZG 15547458 IC50 = 380 nM T38338 C9MRO8 15547459 IC50 = 760 nM T38338 C5O7UI 15547460 IC50 = 5600 nM T38338 CGX0U2 15547461 IC50 = 1300 nM T38338 C8PB4L 15547462 IC50 = 880 nM T38338 C5GUM7 15547463 IC50 = 500 nM T38338 CLF28U 15870889 IC50 = 1300 nM T38338 CPCZ62 16040329 IC50 > 10000 nM T38338 CGD3M1 16659193 IC50 = 730 nM T38338 CEP82X 21076697 IC50 = 2000 nM T38338 C3Y2EQ 21076739 IC50 = 15000 nM T38338 CSZG64 21076740 IC50 = 2600 nM T38338 CFID83 21076741 IC50 = 1600 nM T38338 CN65PY 21076759 IC50 = 2300 nM T38338 CGE0Z3 21076780 IC50 = 5400 nM T38338 CWH9V4 21076782 IC50 = 3800 nM T38338 CKX2Y6 21076784 IC50 = 3400 nM T38338 CQH6N0 21076785 IC50 = 3300 nM T38338 C23DQX 21076786 IC50 = 3400 nM T38338 C3DLY9 21076805 IC50 = 390 nM T38338 C6ZST1 21352112 IC50 = 500 nM T38338 CUKJ32 21352113 IC50 = 370 nM T38338 C8WAT0 21352117 IC50 = 660 nM T38338 CA4F6O 21352149 IC50 = 380 nM T38338 CR7XF5 22084904 IC50 = 7000 nM T38338 C1R3MO 22949255 IC50 = 790 nM T38338 CY2LJ9 22949256 IC50 = 37000 nM T38338 CJ32UX 22949257 IC50 = 680 nM T38338 C32JXL 22949263 IC50 = 6200 nM T38338 C9TA6D 22949266 IC50 = 890 nM T38338 C9SRU6 22949268 IC50 = 28000 nM T38338 C93YKW 22949273 IC50 = 3900 nM T38338 CTR35D 22949275 IC50 = 1500 nM T38338 CUQ94K 22949278 IC50 = 1000 nM T38338 C5AGE4 22949289 IC50 = 37000 nM T38338 C3EL6W 22949292 IC50 = 24000 nM T38338 CXB3Q7 22949294 IC50 = 21000 nM T38338 CLCI39 22949296 IC50 = 1800 nM T38338 C6A7BM 22949298 IC50 = 2000 nM T38338 CAF59B 22949304 IC50 = 1300 nM T38338 CP1HE2 22949305 IC50 = 11000 nM T38338 CA4Z0M 22949307 IC50 = 1700 nM T38338 C2ZJV6 22949308 IC50 = 4600 nM T38338 CV42RZ 23293552 IC50 = 430 nM T38338 CM84OV 23641511 IC50 = 380 nM T38338 C3GY4C 23641891 IC50 = 27 nM T38338 C9WSK4 23642165 IC50 = 560 nM T38338 CI7W3Z 23642174 IC50 = 670 nM T38338 C4WCA6 23642175 IC50 = 460 nM T38338 CVXO48 25101067 IC50 = 1150 nM T38338 CRG10W 25101216 IC50 = 1170 nM T38338 C82FYM 25101375 IC50 = 520 nM T38338 CBIJ72 25101376 IC50 = 190 nM T38338 C2MVC7 25101377 IC50 = 660 nM T38338 CN65YX 25101527 IC50 = 540 nM T38338 CJQ76O 25101676 IC50 = 870 nM T38338 CI39OW 25190761 EC50 < 100000 nM T38338 C53PTZ 25256089 IC50 = 92 nM T38338 C5L7WJ 44269186 IC50 = 780 nM T38338 C6MGI8 44269196 IC50 = 1600 nM T38338 CAL70Z 44269204 IC50 = 320 nM T38338 CF0SG1 44269225 IC50 = 1500 nM T38338 C3QA5J 44269230 IC50 = 490 nM T38338 C25ZPS 44269231 IC50 = 1000 nM T38338 C72CMS 44269232 IC50 = 830 nM T38338 C5E8XB 44269240 IC50 = 320 nM T38338 C4P2ZX 44269249 IC50 = 1000 nM T38338 CVNZ75 44269250 IC50 = 1100 nM T38338 CGNU75 44269268 IC50 = 370 nM T38338 C3OR5G 44269270 IC50 = 400 nM T38338 CYAV72 44269285 IC50 = 300 nM T38338 CL21FU 44296400 IC50 = 500 nM T38338 CU60CQ 44296401 IC50 = 90 nM T38338 C4G9QM 44296746 IC50 = 1200 nM T38338 CC6B3Q 44296747 IC50 = 1000 nM T38338 CAB3K7 44296748 IC50 = 310 nM T38338 CZ1J6X 44296780 IC50 = 440 nM T38338 CEK1J2 44296781 IC50 = 320 nM T38338 CJ0V1N 44296815 IC50 = 420 nM T38338 CDQL42 44296816 IC50 = 270 nM T38338 C8I9BJ 44296817 IC50 = 310 nM T38338 C1FAH0 44305178 IC50 = 26000 nM T38338 CLG30B 44305340 IC50 = 950 nM T38338 C1NJR3 44305341 IC50 = 610 nM T38338 C7KH8Z 44305379 IC50 = 4000 nM T38338 CGF76H 44305380 IC50 = 1800 nM T38338 CX43HP 44305382 IC50 = 1200 nM T38338 C3HC5Q 44308318 IC50 = 1700 nM T38338 CAN9K3 44308319 IC50 = 230 nM T38338 CUQW91 44308346 IC50 = 700 nM T38338 CW0YT6 44308347 IC50 = 560 nM T38338 CQFE28 44308374 IC50 = 36 nM T38338 CZI7U2 44308464 IC50 = 500 nM T38338 C7JM4X 44308465 IC50 = 1700 nM T38338 C6ZMW4 44308753 IC50 = 1000 nM T38338 C7L2FO 44308754 IC50 = 280 nM T38338 C4AW7K 44308756 IC50 = 360 nM T38338 CW1Q0K 44308758 IC50 = 1600 nM T38338 C13HJQ 44308775 IC50 = 130 nM T38338 CR5OD7 44308776 IC50 = 1000 nM T38338 CBG86Z 44308777 IC50 = 1900 nM T38338 CF56XY 44312857 IC50 = 140 nM T38338 CI5ZS2 44312860 IC50 = 150 nM T38338 C2NS4P 44317258 IC50 = 4800 nM T38338 C98ZAH 44317269 IC50 = 2500 nM T38338 CH9VW2 44317301 IC50 > 100000 nM T38338 C2R3GW 44317514 IC50 = 35000 nM T38338 C9K2RP 44317551 IC50 = 15000 nM T38338 CZ95WR 44317565 IC50 = 10000 nM T38338 CO83QZ 44317566 IC50 = 5100 nM T38338 C10CMJ 44317567 IC50 = 1100 nM T38338 CE4MJ0 44317613 IC50 = 7400 nM T38338 CJE76X 44382868 IC50 = 5800 nM T38338 C41HKO 44382869 IC50 = 400 nM T38338 CIP6F5 44382871 IC50 = 920 nM T38338 C7BXI8 44382916 IC50 = 1200 nM T38338 C9VQ3L 44383000 IC50 = 390 nM T38338 CG5BQ1 44383003 IC50 = 120 nM T38338 CIF26H 44383007 IC50 = 380 nM T38338 CN9KH1 44383009 IC50 = 1300 nM T38338 CZ05CO 44383016 IC50 = 330 nM T38338 CFWB96 44383017 IC50 = 360 nM T38338 C2A8CQ 44383059 IC50 = 1500 nM T38338 CLV04D 44383125 IC50 = 6400 nM T38338 CAH17S 44383185 IC50 = 720 nM T38338 CSJZ21 44383237 IC50 = 120 nM T38338 C1ARI8 44383291 IC50 = 2300 nM T38338 CJF7X3 44383300 IC50 = 2800 nM T38338 CL1V5I 44383331 IC50 = 500 nM T38338 C7AP4V 44383354 IC50 = 1400 nM T38338 CBS07P 44383446 IC50 = 3800 nM T38338 CP0YD3 44383450 IC50 = 200 nM T38338 CS5DM6 44383882 IC50 = 3100 nM T38338 CT03BS 44383921 IC50 = 2300 nM T38338 CSOX95 44383978 IC50 = 280 nM T38338 CA8LX4 44384087 IC50 = 2200 nM T38338 CB05DS 44384089 IC50 = 4400 nM T38338 C5UE3M 44384194 IC50 = 880 nM T38338 C4SML2 44384244 IC50 = 610 nM T38338 C3SDG2 44384250 IC50 = 600 nM T38338 CV7F4K 44384252 IC50 = 1900 nM T38338 C0S3TA 44384260 IC50 = 350 nM T38338 CK8CO5 44384319 IC50 = 610 nM T38338 C7LC2M 44384434 IC50 = 2700 nM T38338 C5IZ6N 44386758 IC50 = 1800 nM T38338 CMD79Z 44397141 IC50 = 3000 nM T38338 CRS05Y 44407306 IC50 = 2900 nM T38338 C37QCG 44407322 IC50 = 10000 nM T38338 C7N2YF 44407404 IC50 = 830 nM T38338 CFQX34 44407458 IC50 = 1000 nM T38338 CGX29Y 44430888 IC50 = 2410 nM T38338 CP3IK9 44430890 IC50 = 1340 nM T38338 C34KHL 44430891 IC50 = 1290 nM T38338 C36KRI 44430892 IC50 = 8130 nM T38338 C3BL8H 44430893 IC50 = 29800 nM T38338 CRUM21 44430899 IC50 = 1300 nM T38338 CFTE23 44430918 IC50 = 3970 nM T38338 CC47KR 44430919 IC50 = 4420 nM T38338 CYB50Z 44430922 IC50 = 580 nM T38338 C8RCK2 44430923 IC50 = 4150 nM T38338 C3OZY5 44430926 IC50 = 1400 nM T38338 C13ZHV 44430928 IC50 = 590 nM T38338 CL4TS6 44430930 IC50 = 1260 nM T38338 C37RQE 44430932 IC50 = 4920 nM T38338 CS68OF 44430933 IC50 = 8930 nM T38338 CBDP46 44430935 IC50 = 1960 nM T38338 C4K6IB 44430936 IC50 = 560 nM T38338 C74DCW 44430937 IC50 = 770 nM T38338 C41CXK 44460427 IC50 = 400 nM T38338 C6AR7Z 44460428 IC50 = 690 nM T38338 CZRD12 44460429 IC50 = 670 nM T38338 C7ER3L 44460430 IC50 = 190 nM T38338 CEQ5Y1 44460714 IC50 = 1800 nM T38338 CMF9Y5 44460732 IC50 = 1000 nM T38338 CV51KN 44460792 IC50 = 14000 nM T38338 C8M4LG 44460793 IC50 = 17000 nM T38338 C6B9GZ 44460817 IC50 = 1800 nM T38338 CNCM23 44461078 IC50 = 1800 nM T38338 CG6ZI0 44461093 IC50 = 290 nM T38338 CLK98B 44461094 IC50 = 120000 nM T38338 C9D5QG 44461096 IC50 = 2200 nM T38338 C7X6ZQ 44461108 IC50 = 1100 nM T38338 C8UKM3 44461109 IC50 = 490 nM T38338 CSG28K 44461117 IC50 = 1100 nM T38338 C19ZCY 46861765 IC50 = 28710 nM T38338 CUDE92 50898773 IC50 = 4900 nM T38338 C90UKY 50899643 IC50 > 10000 nM T38338 CPS12B 53317097 IC50 > 30000 nM T38338 CB03RY 53317952 IC50 = 880 nM T38338 CM0LP8 53317953 IC50 = 680 nM T38338 CT05AO 53323237 IC50 = 600 nM T38338 C09GHY 57580315 IC50 = 710 nM T38338 C7BDI5 57580339 IC50 = 450 nM T38338 CPUZ69 59447115 IC50 = 510 nM T38338 CHK0J5 59447390 IC50 = 360 nM T38338 C0M9KS 66590257 IC50 = 851.14 nM T38338 CXS5D6 66590299 IC50 = 1862.09 nM T38338 C26SJE 66590331 IC50 = 457.09 nM T38338 C5D4VT 66590464 IC50 = 741.31 nM T38338 CH5YQ8 66590494 IC50 = 870 nM T38338 C4YB5I 66590600 IC50 = 1510 nM T38338 CD57QH 66590630 IC50 = 520 nM T38338 C0CLT7 66590943 IC50 = 1047.13 nM T38338 CK06BS 66590948 IC50 = 2818.38 nM T38338 CTP46W 66591036 IC50 = 770 nM T38338 CX1WY2 66591069 IC50 = 1890 nM T38338 C0I9ML 66591354 IC50 = 960 nM T38338 C0JX1S 66996537 IC50 = 1230.27 nM T38338 C7Z8IA 66997369 IC50 = 5150 nM T38338 CMK42I 66997462 IC50 = 1174.9 nM T38338 C9UGC7 68573974 IC50 = 490 nM T38338 CTH21S 69472592 EC50 = 14230 nM T38338 C05FUX 71450594 EC50 = 11290 nM T38338 C05HLQ 71452434 EC50 = 30020 nM T38338 CLI8A4 71452435 EC50 > 100000 nM T38338 CAWK20 71452436 EC50 > 1000000 nM T38338 CWE64K 71453870 IC50 = 2500 nM T38338 CN1QD3 71454199 EC50 > 1000000 nM T38338 CET6W1 71455597 IC50 = 370 nM T38338 CLB0V3 71455942 EC50 > 100000 nM T38338 CJ5NC0 71455943 EC50 > 100000 nM T38338 C5GO3U 71455944 EC50 > 100000 nM T38338 CN13QL 71457386 IC50 = 240 nM T38338 C0S8PA 71457387 IC50 = 660 nM T38338 CTK62I 71457748 EC50 > 100000 nM T38338 CJ3I7G 71457749 EC50 > 1000000 nM T38338 CZ09XC 71459652 EC50 > 100000 nM T38338 C9M5ES 71459653 EC50 > 100000 nM T38338 C9AB7D 71459654 EC50 > 100000 nM T38338 C3O1QA 71459655 EC50 > 100000 nM T38338 CBQ86V 71459656 EC50 > 100000 nM T38338 C6HKD3 71459657 EC50 > 100000 nM T38338 C6D8HC 71459658 EC50 > 100000 nM T38338 CD98PK 71461022 IC50 = 1100 nM T38338 CEC98W 71461024 IC50 = 60 nM T38338 CN17SY 71461025 IC50 = 120 nM T38338 C2T0OS 71461386 EC50 > 100000 nM T38338 CLT7E6 71461387 EC50 > 70000 nM T38338 C2WZB4 71462748 IC50 = 300 nM T38338 CSE6Z5 71463101 EC50 = 7210 nM T38338 CE2F1M 71463102 EC50 > 100000 nM T38338 CSR18T 71463103 EC50 > 100000 nM T38338 C9Q7YL 71463104 EC50 > 100000 nM T38338 CX24MZ 71463105 EC50 > 100000 nM T38338 C8Q7IC 71819113 IC50 = 790 nM T38338 C0M9XZ 71819114 IC50 = 860 nM T38338 C5TI0Y 71819115 IC50 = 389.05 nM T38338 CL9P4V 72301648 IC50 = 88 nM T38338 C7B6JU 72543966 IC50 = 340 nM T38338 C5XS4J 72544205 IC50 = 370 nM T38338 C0WTY6 72544206 IC50 = 970 nM T38338 CB59MH 72544207 IC50 = 470 nM T38338 C2GVQ0 73291871 IC50 = 30 nM T38338 COY30K 73291874 IC50 = 2 nM T38338 CN26XA 73291875 IC50 = 3 nM T38338 CRF4K3 73292224 IC50 = 7 nM T38338 C6SHE2 73292225 IC50 = 12 nM T38338 CKA79H 73292924 IC50 = 1 nM T38338 C6EW5M 73292925 IC50 = 1 nM T38338 CN2BS7 73293096 IC50 = 29 nM T38338 CY6J7T 73293610 IC50 = 11 nM T38338 C6FLS3 73293612 IC50 = 6 nM T38338 CP4IT3 73293983 IC50 = 3 nM T38338 CYS8H4 73294550 IC50 = 7 nM T38338 CGJC94 73294553 IC50 = 1 nM T38338 C02XJO 76313667 IC50 = 760 nM T38338 CZ5NL6 76317170 IC50 = 380 nM T38338 CQN91E 76324551 IC50 = 290 nM T38338 CQ4S7V 76324552 IC50 = 430 nM T38338 C6XY5G 76328112 IC50 = 48 nM T38338 CWJ65U 76331788 IC50 = 21 nM T38338 C9CTQ0 76331789 IC50 = 48 nM T38338 C4OXA6 76331790 IC50 = 390 nM T38338 CP42DU 76331791 IC50 = 190 nM T38338 C5VW7X 76331792 IC50 = 270 nM T38338 CQ15FV 76331793 IC50 = 310 nM T38338 CV6KW2 76335376 IC50 = 350 nM T38338 CWCU76 76335377 IC50 = 72 nM T38338 CN10FE 90040082 IC50 = 20 nM T38338 CDBZ84 90200902 IC50 = 2 nM T38338 CKTF80 90201263 IC50 = 44 nM T38338 CL15MQ 122189314 IC50 = 6700 nM T38338 C1PRY5 122189316 IC50 = 4300 nM T38338 C4EF6B 122189318 IC50 = 5900 nM T38338 CX35ZS 122189320 IC50 = 9400 nM T38338 CZ16JP 122189321 IC50 = 9500 nM T38338 CEF2Z5 136186016 IC50 = 35000 nM T38338 CGV18I 145967628 IC50 = 77000 nM T38338 CQ74PV 145967661 IC50 = 105000 nM T38338 C7Y0MU 145967892 IC50 = 98000 nM T38338 CE3GA1 145968071 IC50 = 49000 nM T38338 C5YK7S 145968281 IC50 = 202000 nM T38338 C09HME 145968567 IC50 = 244000 nM T38338 C53KZP 145968632 IC50 = 59000 nM T38338 CM06JK 145968873 IC50 = 51000 nM T38338 CTE5M6 145968992 IC50 = 130000 nM T38338 C0RFY3 145969009 IC50 = 103000 nM T38338 C7KCA4 145969044 IC50 = 46000 nM T38338 CFV2D8 145969191 IC50 = 205000 nM T38338 C3PN7K 145969264 IC50 = 65000 nM T38338 CJ4BF6 145969488 IC50 = 432000 nM T38338 CG56AM 145969886 IC50 = 253000 nM T38338 C9SQV7 145969924 IC50 = 283000 nM T38338 CKX32N 145970126 IC50 = 167000 nM T38338 CXNE63 145970149 IC50 = 143000 nM T38338 C4XD2J 145970156 IC50 = 185000 nM T38338 C3AR7T 145970259 IC50 = 106000 nM T38338 C0V7HM 145970794 IC50 = 144000 nM T38338 CD9SA3 145970877 IC50 = 40000 nM T38338 CL9ZA4 145971033 IC50 = 117000 nM T38338 CLQ74T 145971053 IC50 = 100000 nM T38338 C5LCQ7 145971063 IC50 = 113000 nM T38338 CE9P1Z 145971143 IC50 = 69000 nM T38338 C7CUB1 145984146 IC50 = 28 nM T38338 C98BZP 145986355 IC50 = 41000 nM T38338 C2YU5X 145988084 IC50 = 22 nM T38338 C4NP8S 145988617 IC50 = 218000 nM T38338 CA2XP0 145988629 IC50 = 368000 nM T38338 D07ADR 2422 EC50 > 1000000 nM T38338 D07BDQ 44356037 IC50 = 320 nM T38338 D08RJC 44460434 IC50 = 970 nM T38338 D0C3VI 44356550 IC50 = 590 nM T38338 D0FF6S 16038374 IC50 > 10000 nM T38338 D0PE8P 9916734 IC50 = 40 nM T38338 D0UB0T 9823703 IC50 = 1500 nM T38338 D0Y0ES 3707 EC50 > 1000000 nM T57316 CW9Z0M 10405091 IC50 = 8.9 ug.mL-1 T57316 CX8OR6 11080475 IC50 = 48.5 ug.mL-1 T57316 CY0NO4 11248738 IC50 = 1000 nM T57316 C2RFL1 44315263 Ki = 1600 nM T57316 C5O2KR 44315516 Ki = 253000 nM T57316 CCH8V0 44315557 IC50 = 400000 nM T57316 CM8O4K 44337239 IC50 = 72.5 ug.mL-1 T57316 CELN92 44337250 IC50 = 10.2 ug.mL-1 T57316 CJ2Y8U 44337258 IC50 > 100 ug.mL-1 T57316 D06PRC 5281650 IC50 = 46.5 ug.mL-1 T27861 D0A3ZU 134780 IC50 = 1200 nM T27861 D0Q5NX 216326 IC50 = 1500 nM T27861 D0U7GK 5426 Ki = 22700 nM T27861 D01XVX 67335295 IC50 = 60 nM T27861 CR81TN 6213 Ki = 137490000 nM T27861 C1BH2K 11439 Ki = 26200 nM T27861 CX85GI 70726 Ki = 103100 nM T27861 CQ63YN 71020635 IC50 > 10 nM T27861 CWCV69 131988640 IC50 = 5.5 nM T27861 C9XB0W 139600332 IC50 = 2 nM T52067 D00HWO 19003 Ki = 43651.58 nM T52067 D01PLN 6024 Ki = 8300000 nM T52067 D04KTZ 6098 Ki = 950000 nM T52067 D05UBX 42008 Ki = 4265795.19 nM T52067 D06OVY 5362065 Ki = 2570395.78 nM T52067 D06YHL 456255 Ki = 2800000 nM T52067 D0A1CB 5479537 Ki = 10964781.96 nM T52067 D0D1HA 5742673 Ki = 19952623.15 nM T52067 D0F6EO 33613 Ki = 426579.52 nM T52067 D0MB8I 6196 Ki = 3300000 nM T52067 D0PW7C 51039 Ki = 28840.32 nM T52067 D0R2KJ 18381 Ki = 416869.38 nM T52067 D0W6CA 6335986 Ki = 30902954.33 nM T52067 D0X9ZC 47965 Ki = 3000 nM T52067 D0Y2IE 5479529 Ki = 12589254.12 nM T52067 D0YA9Z 6249 Ki = 1288249.55 nM T52067 D0Z5EM 27447 Ki = 75000 nM T52067 D00QAR 5904 Ki = 10964781.96 nM T52067 D0F8IO 5773 Ki = 8500000 nM T52067 CXY67D 11163 Ki = 53703.18 nM T52067 CD6FT7 70910 Ki = 18000 nM T52067 CDO2S7 73587 Ki = 3090295.43 nM T52067 C7YC2T 80817 Ki = 10000 nM T52067 C5F9KD 83525 Ki = 12000 nM T52067 CTV32A 88656 Ki = 794.33 nM T52067 CS28ZP 96796 Ki = 269153.48 nM T52067 CPGC40 97050 Ki = 10964781.96 nM T52067 C35FZA 194260 Ki = 2570395.78 nM T52067 C47QLZ 439360 Ki = 128824.96 nM T52067 C5ZW4M 439498 Ki = 28840.32 nM T52067 CW9JK0 471583 Ki = 150000 nM T52067 C4HCS7 1549433 Ki = 6000 nM T52067 CUN54L 1549453 Ki = 30902.95 nM T52067 CQ6IO0 1551643 Ki = 3467.37 nM T52067 CT5W1J 3082062 Ki = 1995.26 nM T52067 CNRG81 5361871 Ki = 8912509.38 nM T52067 CM47TY 5478845 Ki = 18000 nM T52067 CJHI21 5484352 Ki = 6000 nM T52067 C6C1TR 5488196 Ki = 15848.93 nM T52067 CF07VG 5496455 Ki = 4365.16 nM T52067 CG30YS 6713928 Ki = 724435.96 nM T52067 C6KTO7 6992304 Ki = 14000 nM T52067 C9W1MN 6992506 Ki = 30000 nM T52067 CKED87 6993082 Ki = 3000 nM T52067 C04HTR 6993090 Ki = 37000 nM T52067 CK3Q0Z 6993120 Ki = 3800 nM T52067 CY4FN2 6993401 Ki = 3981.07 nM T52067 C7HIQ9 6998029 Ki = 7000 nM T52067 CMB48H 7009555 Ki = 2500 nM T52067 CVI1B7 7009579 Ki = 7000 nM T52067 CXH50C 7009600 Ki = 8912.51 nM T52067 C15XOM 7010504 Ki = 40738.03 nM T52067 CA2XY3 7016106 Ki = 22908.68 nM T52067 C71EGJ 7021452 Ki = 12000 nM T52067 C2PR6I 7023107 Ki = 38904.51 nM T52067 CHY42A 7079450 Ki = 2089296.13 nM T52067 C28NMU 7408195 Ki = 7943.28 nM T52067 C70ZHW 7408741 Ki = 891250.94 nM T52067 CVP24W 9818200 Ki = 22908.68 nM T52067 CDO9J0 9837272 Ki = 38904.51 nM T52067 CP7C8K 9838453 Ki = 158489.32 nM T52067 CV7Z4H 10159368 Ki = 1698.24 nM T52067 C3WV9X 11223118 Ki = 14000 nM T52067 CBR19W 20112139 Ki = 15848.93 nM T52067 C5HXU3 23675312 Ki = 11100000 nM T52067 C2OEG0 40496728 Ki = 6000 nM T52067 CMR2Y1 44398488 Ki = 8912.51 nM T52067 CX3SC4 44398561 Ki = 300 nM T52067 CAIY06 56665053 Ki = 549540.87 nM T52067 CJKO83 56668511 Ki = 239883.29 nM T52067 CU6YH8 56682043 Ki = 190000 nM T52067 CX08JM 56682044 Ki = 6000 nM T52067 CY50OA 56682045 Ki = 109647.82 nM T52067 D0A1PW 11579 Ki = 229086.77 nM T89360 D06IAR 60961 Ki > 100000 nM T89360 D0F0ZE 153241 IC50 = 10 nM T89360 CEA89F 10256 IC50 = 22700 nM T89360 C8IOM3 230282 IC50 = 20900 nM T89360 C5ZC0A 497770 IC50 = 20 nM T89360 C4U0OC 497771 IC50 = 25 nM T89360 CLO3N7 497772 IC50 = 70 nM T89360 C4A6KW 497773 IC50 = 85 nM T89360 C0O2NT 497774 IC50 = 23 nM T89360 C2Z5CN 497775 IC50 = 97 nM T89360 CI1L3Y 497776 IC50 = 115 nM T89360 CG2VI5 497777 IC50 = 127 nM T89360 CBD46Q 497781 IC50 = 27 nM T89360 C15XDV 497782 IC50 = 86 nM T89360 CZ8C9D 497783 IC50 = 30 nM T89360 CPJZ06 497784 IC50 = 18 nM T89360 CY06OL 497785 IC50 = 22 nM T89360 CE3SV8 497786 IC50 = 15 nM T89360 C9O4ES 497787 IC50 = 17 nM T89360 C19KSA 497788 IC50 = 13 nM T89360 C6V0PS 497790 IC50 = 11 nM T89360 C25GVM 497791 IC50 = 13 nM T89360 C1RCH0 497792 IC50 = 12 nM T89360 CSR10C 510912 IC50 = 19 nM T89360 C5NK2J 510914 IC50 > 10000000 nM T89360 CMH8E2 510915 IC50 = 670 nM T89360 CRA21X 510916 IC50 = 230 nM T89360 CZU3J2 510917 IC50 > 5000000 nM T89360 C42PBY 510918 IC50 = 33 nM T89360 C85EAF 510919 IC50 = 440 nM T89360 C8S1IN 510920 IC50 = 490 nM T89360 CTG6D2 510921 IC50 > 550 nM T89360 CFM70Y 510923 IC50 = 280 nM T89360 C8WB2K 510924 IC50 = 180 nM T89360 CZK7N2 510925 IC50 = 260 nM T89360 C7BXI5 510926 IC50 = 200 nM T89360 CT78CW 510927 IC50 = 130 nM T89360 CH65RZ 510928 IC50 = 100 nM T89360 C89EVQ 510929 IC50 = 94 nM T89360 CDX01M 510930 IC50 = 180 nM T89360 CTA12W 510933 IC50 = 240 nM T89360 CY8NB9 510934 IC50 = 420 nM T89360 CZ8B4H 510935 IC50 = 210 nM T89360 CA8V3T 588991 IC50 > 5000 nM T89360 C0BCA8 612046 IC50 > 5000 nM T89360 C1K4GB 675297 IC50 >= 5000 nM T89360 C8WTH9 776662 IC50 >= 5000 nM T89360 COJ29X 890649 IC50 = 2100 nM T89360 CQC02U 1139867 IC50 > 5000 nM T89360 CLQ93F 1256741 IC50 > 5000 nM T89360 CO48PU 1367213 IC50 > 5000 nM T89360 CUK93P 2309238 IC50 >= 5000 nM T89360 CK47YQ 2336594 IC50 >= 5000 nM T89360 CM2G8F 2349729 IC50 > 5000 nM T89360 C7TZ5D 2930546 IC50 = 5700 nM T89360 C9A5GP 2953497 IC50 > 5000 nM T89360 CC69EB 2953546 IC50 > 5000 nM T89360 CS1OL3 2990648 IC50 > 5000 nM T89360 C70OXL 3006288 Ki = 3000 nM T89360 CF8N3B 3140491 EC50 > 50000 nM T89360 CAY86S 3312427 IC50 = 2100 nM T89360 CC7WN4 3984960 IC50 > 5000 nM T89360 C0CX1O 4084632 IC50 > 5000 nM T89360 C7KV2M 5173303 IC50 > 5000 nM T89360 CIXQ25 6478685 IC50 = 1400 nM T89360 CW62YA 6479888 IC50 = 790 nM T89360 CN29OD 6618978 IC50 > 50000 nM T89360 CQ96MK 9400179 IC50 > 5000 nM T89360 C75FLA 9797026 IC50 = 10 nM T89360 CND1O9 9797707 IC50 = 190 nM T89360 CJ29KX 9798978 IC50 = 47 nM T89360 C6KM5A 9817941 IC50 = 18.6 nM T89360 CW84FQ 9819013 IC50 = 19 nM T89360 CWC79A 9822362 IC50 < 5 nM T89360 CI8K7N 9838854 IC50 = 5 nM T89360 CLIF21 9842306 IC50 = 23 nM T89360 C0TUD2 9856426 IC50 = 110 nM T89360 CM73SE 9858793 IC50 < 5 nM T89360 CRLZ80 9878581 IC50 = 220 nM T89360 CGB78L 9880305 IC50 = 9 nM T89360 CW3S9G 9883477 Ki = 7 nM T89360 C0S2OY 9884816 IC50 > 10000 nM T89360 CKY2D7 9901690 IC50 = 55 nM T89360 CW4DN6 9906308 IC50 = 150 nM T89360 CG16TY 9907596 IC50 = 30 nM T89360 C64CDR 9912093 IC50 = 20 nM T89360 C4B2QY 9913339 IC50 = 17 nM T89360 CWR2S7 9921131 IC50 = 300 nM T89360 C7HBG3 9921906 IC50 = 200 nM T89360 CK13BM 9923286 IC50 = 63 nM T89360 C5LZ0F 9939667 IC50 = 2600 nM T89360 CO6CV0 9946220 IC50 = 1500 nM T89360 C2H4YG 9947722 IC50 = 14 nM T89360 C4F9QU 9949504 IC50 = 240 nM T89360 CYOD07 9949676 IC50 = 52 nM T89360 CYU51P 9966370 IC50 = 32 nM T89360 CV68RP 9966794 IC50 = 70 nM T89360 CN59SI 9976927 IC50 = 300 nM T89360 CNU0B4 10113643 IC50 < 5 nM T89360 CYM8X2 10117522 IC50 = 68 nM T89360 CI06PF 10126668 IC50 = 130 nM T89360 C49BEK 10131333 IC50 = 34 nM T89360 CG53VS 10131739 IC50 = 18 nM T89360 C0XAE4 10131741 IC50 = 320 nM T89360 C3G5HN 10134808 IC50 = 12 nM T89360 CA6V7K 10135675 IC50 = 55 nM T89360 C9G7LN 10136663 IC50 = 16 nM T89360 CUA05R 10136713 IC50 = 14 nM T89360 CLN19D 10159708 IC50 = 18 nM T89360 C6ELS3 10164678 IC50 = 18 nM T89360 CF9X7W 10172305 IC50 = 86 nM T89360 C2T1ZL 10177736 IC50 = 30 nM T89360 C7Y0NW 10180910 IC50 = 13 nM T89360 CE6F2O 10182966 IC50 = 12 nM T89360 C2O5AZ 10194459 IC50 = 390 nM T89360 CS7W5A 10200804 IC50 = 22 nM T89360 C7MY4A 10203029 IC50 = 15 nM T89360 CR1N6A 10215650 IC50 = 57 nM T89360 CQT82I 10221809 IC50 = 25 nM T89360 CR59ZE 10225421 IC50 = 20 nM T89360 C2X6TP 10233633 Ki = 380 nM T89360 CN4V6E 10236318 IC50 = 104 nM T89360 C05NVJ 10259194 Ki = 300 nM T89360 CW49NI 10269167 IC50 = 2200 nM T89360 CK4L2E 10269960 IC50 = 1100 nM T89360 C87NBG 10270744 IC50 = 28 nM T89360 C48IXR 10273163 IC50 = 6 nM T89360 CN0CM7 10276405 IC50 < 5 nM T89360 CC7PU9 10292172 IC50 = 280 nM T89360 C5OGE6 10297318 IC50 = 11 nM T89360 CLO3B8 10309152 IC50 = 188 nM T89360 CD4L2P 10309428 IC50 = 160 nM T89360 CGF36N 10315709 IC50 < 5 nM T89360 C7IQE9 10323922 IC50 = 16 nM T89360 CV7RA9 10338010 IC50 = 400 nM T89360 CH74QD 10345767 IC50 = 40 nM T89360 CO3GQ6 10358016 IC50 = 28 nM T89360 CU8C2Y 10358687 IC50 = 57 nM T89360 CNG97X 10361468 IC50 = 440 nM T89360 C5WXT0 10381198 IC50 = 12.6 nM T89360 COT86A 10412176 IC50 = 58 nM T89360 CDXB75 10434905 IC50 = 7 nM T89360 C49WRJ 10462123 IC50 = 700 nM T89360 C28SEY 10492850 IC50 = 51800 nM T89360 CF3D8K 10495354 IC50 = 33.5 nM T89360 C7BS3V 10495605 IC50 = 8.51 nM T89360 C02SWN 10496064 IC50 = 465 nM T89360 C6GK2Y 10497453 IC50 = 1800 nM T89360 C0MRX3 10515627 IC50 > 100000 nM T89360 C6MY4S 10518087 IC50 = 537 nM T89360 CPC4F9 10519658 IC50 = 244 nM T89360 CC3HM6 10519938 IC50 = 184 nM T89360 CB5SI1 10544613 IC50 = 231 nM T89360 C7KPV1 10546858 IC50 = 130 nM T89360 C8M9IK 10566972 IC50 = 1700 nM T89360 C37FNC 10567307 IC50 = 437 nM T89360 CFN5V6 10568712 IC50 = 644 nM T89360 CXMB45 10569189 IC50 = 795 nM T89360 C8WM7C 10590744 IC50 = 515 nM T89360 CV4A8H 10593915 IC50 > 100000 nM T89360 C0AWD9 10616470 IC50 = 557 nM T89360 CXE6C1 10637391 IC50 = 959 nM T89360 C06DYP 10643207 IC50 = 1040 nM T89360 C71JXF 10652408 Ki = 270 nM T89360 C2S6QL 10662964 IC50 = 2880 nM T89360 C1CFT4 10663129 IC50 = 15500 nM T89360 CUGI51 10682843 IC50 = 90800 nM T89360 C56XFB 10685057 IC50 = 50000 nM T89360 C50IUC 10686776 IC50 = 11800 nM T89360 CR0MC9 10687933 IC50 > 100000 nM T89360 C5H9AV 10688491 IC50 = 763 nM T89360 CDY41T 10709084 IC50 = 69.3 nM T89360 CMV3K1 10709184 IC50 = 1380 nM T89360 C1S4LW 10709494 IC50 = 14800 nM T89360 C1N0ZQ 10709767 IC50 = 1120 nM T89360 CA7IP0 10709955 IC50 = 52300 nM T89360 CEI9K7 10710928 IC50 = 681 nM T89360 CSW57G 10711760 IC50 = 410 nM T89360 C9S8WO 10713240 IC50 = 462 nM T89360 C87BPJ 10732226 IC50 = 6960 nM T89360 CA4L7V 10735580 IC50 = 126 nM T89360 C0PL3X 10735599 IC50 = 121 nM T89360 CLYM27 10746991 Ki = 320 nM T89360 C8A4YB 10756343 IC50 = 1080 nM T89360 CTSY82 10757447 IC50 = 489 nM T89360 CA4S3R 10758796 IC50 = 50.7 nM T89360 COG9Z8 10759053 IC50 > 100000 nM T89360 C39CHI 10759638 IC50 = 620 nM T89360 CR2A8D 10780300 IC50 = 18800 nM T89360 C1RX9K 10782926 IC50 = 420 nM T89360 C0IM7L 10787380 IC50 = 592 nM T89360 CB4YR2 10803200 IC50 = 1600 nM T89360 CSCY60 10804648 IC50 = 1220 nM T89360 CPU5G1 10805499 IC50 = 140 nM T89360 C9ZU8R 10826397 IC50 = 17000 nM T89360 CR83PV 10826452 IC50 > 100000 nM T89360 C5WAI9 10828540 IC50 = 289 nM T89360 CJ4S2P 10832148 IC50 = 36.7 nM T89360 CDT59Z 10841975 Ki = 57900 nM T89360 CB92AM 10851956 IC50 = 534 nM T89360 C0OIC1 10852317 IC50 = 11900 nM T89360 CQHG03 10872836 IC50 = 104 nM T89360 CO1V7B 10896057 IC50 = 20 nM T89360 C9KVM0 10927586 IC50 = 141 nM T89360 CT8DX2 11069304 Ki = 400 nM T89360 CD4JG6 11118869 IC50 = 254 nM T89360 CAL6D3 11162210 IC50 >= 5000 nM T89360 CR5J2F 11440390 IC50 = 13 nM T89360 C0US3F 11670037 IC50 = 35 nM T89360 C3XHB6 11674857 IC50 = 76 nM T89360 C17DLS 11828231 Ki = 470 nM T89360 C58ZYV 11962096 IC50 = 84 nM T89360 C6IMB3 12093478 IC50 = 970 nM T89360 C54TFI 12093480 IC50 = 110 nM T89360 CGT24F 12093481 IC50 = 73 nM T89360 CLP6T3 15040652 IC50 > 5000 nM T89360 C1N8XS 16007061 IC50 = 13 nM T89360 C4RKU7 16046198 Ki = 37 nM T89360 CKTA70 16484765 IC50 = 2600 nM T89360 CH0R7U 16484780 IC50 = 3200 nM T89360 CN5AB6 16747704 Ki = 18800 nM T89360 C94FVH 16748017 IC50 = 19 nM T89360 C47PSG 16748018 IC50 = 95 nM T89360 CK75MC 16748019 IC50 = 53 nM T89360 CZEQ54 16748020 IC50 = 42 nM T89360 C56GJV 16748021 IC50 = 11 nM T89360 CF85SK 16748022 IC50 = 11 nM T89360 C81DQT 16748142 IC50 = 12 nM T89360 C93QIS 16748143 IC50 = 7.9 nM T89360 C0JYU6 16748144 IC50 = 23 nM T89360 CI3DJ9 16748145 IC50 = 14 nM T89360 CA6M0N 16748267 IC50 = 12 nM T89360 CGSB38 16748274 IC50 = 20 nM T89360 CIC18J 16748525 IC50 = 29 nM T89360 CD57VL 16748526 IC50 = 20 nM T89360 CUQG95 16748527 IC50 = 10 nM T89360 CN1P8T 16748528 IC50 = 17 nM T89360 CYWJ25 16748529 IC50 = 22 nM T89360 CY64OX 16748634 IC50 = 59 nM T89360 CCTY21 16748636 IC50 = 431 nM T89360 C1DU6C 16748637 IC50 = 53 nM T89360 CH5E8D 16748745 IC50 = 11 nM T89360 CT8S1K 17032699 IC50 > 5000 nM T89360 CQT58O 17033137 IC50 > 5000 nM T89360 CS1LN8 17033372 IC50 > 5000 nM T89360 CSU17Z 18184806 IC50 = 400 nM T89360 CUWA47 18467513 IC50 = 380 nM T89360 C3LSH2 19165245 IC50 >= 5000 nM T89360 CZUJ07 19168353 IC50 >= 5000 nM T89360 C7ZL3T 19168356 IC50 >= 5000 nM T89360 CB62FV 20766912 IC50 > 10000 nM T89360 CVR34M 20766928 IC50 > 5000 nM T89360 CTMK79 20766951 IC50 > 10000 nM T89360 CEW1H6 20766964 IC50 > 10000 nM T89360 CF6VY0 21343422 IC50 = 28 nM T89360 CMFZ98 21343423 IC50 = 47 nM T89360 CKBR14 21343449 IC50 = 45 nM T89360 CR8PG0 22058483 IC50 = 200 nM T89360 CJEA25 22058485 IC50 = 170 nM T89360 C82WXQ 22058487 IC50 = 130 nM T89360 CMW8Z1 22058491 IC50 = 74 nM T89360 C9RN7Y 22058493 IC50 = 18 nM T89360 CDN25T 22058495 IC50 = 890 nM T89360 CW59LM 22058498 IC50 = 66 nM T89360 C0N5HJ 22058499 IC50 = 300 nM T89360 CG1ET0 22058500 IC50 = 210 nM T89360 C80VAD 22058504 IC50 > 10000 nM T89360 C50PZT 22058514 IC50 = 630 nM T89360 C2XKA3 22058516 IC50 = 540 nM T89360 CHD96V 22058517 IC50 = 140 nM T89360 CZQ9S0 22058521 IC50 = 260 nM T89360 C1SQF5 22058523 IC50 = 210 nM T89360 CG1XV3 22058530 IC50 = 35 nM T89360 C8QYM5 22058533 IC50 = 110 nM T89360 CFY48L 22058535 IC50 = 130 nM T89360 C98PNG 22058536 IC50 = 870 nM T89360 CQV4C5 22058537 IC50 = 210 nM T89360 CT81BG 22058540 IC50 = 330 nM T89360 C50SZG 22058546 IC50 = 230 nM T89360 CJ0E2N 22058549 IC50 = 410 nM T89360 CUV9T5 22058554 IC50 = 120 nM T89360 CN61PF 22058555 IC50 = 60 nM T89360 C05UQA 22093099 IC50 = 180 nM T89360 CVA2J7 22093112 IC50 = 110 nM T89360 CIEV83 22226545 IC50 > 5000 nM T89360 CO5D4T 22238480 IC50 = 64 nM T89360 C8NFO7 22238485 IC50 = 230 nM T89360 C8Z7YO 22238488 IC50 = 360 nM T89360 C8Z7TF 22238492 IC50 = 130 nM T89360 C4RL8K 22238495 IC50 = 220 nM T89360 CHD0W4 22238496 IC50 = 500 nM T89360 CS4O3X 22349495 IC50 > 1000 nM T89360 C2J8FN 22349571 IC50 = 160 nM T89360 C2E5SM 22459608 IC50 = 41 nM T89360 CF2W6L 22459610 IC50 = 120 nM T89360 C0AF6L 22459619 IC50 = 44 nM T89360 CYBK83 22459624 IC50 = 170 nM T89360 C5BEX9 22459627 IC50 = 110 nM T89360 CP21KX 22459655 IC50 = 190 nM T89360 CMO17X 22459661 IC50 = 410 nM T89360 CG68HF 22459673 IC50 = 54 nM T89360 CDB6I3 22459677 IC50 = 310 nM T89360 C38PCH 22459686 IC50 = 76 nM T89360 C9O4YG 22459693 IC50 = 760 nM T89360 C6PF0W 22459706 IC50 = 32 nM T89360 CK1W8G 22459707 IC50 > 1600 nM T89360 C65GMW 22459716 IC50 = 78 nM T89360 CEJ85U 22459723 IC50 > 5000 nM T89360 CTIL79 22459725 IC50 = 160 nM T89360 C2R1IB 22459727 IC50 = 300 nM T89360 C97UNB 22459730 IC50 = 410 nM T89360 CLK5B2 22459738 IC50 = 330 nM T89360 CSQ68W 22459746 IC50 = 100 nM T89360 C0E7BC 22459748 IC50 = 59 nM T89360 C7BNW0 22459765 IC50 = 130 nM T89360 CIT2G5 22459770 IC50 = 330 nM T89360 C4RI2U 22459775 IC50 > 10000 nM T89360 C5PST6 22459779 IC50 = 41 nM T89360 C0CYK4 22459787 IC50 = 21 nM T89360 CIK04R 22558406 IC50 > 10000 nM T89360 C63IGS 22946285 IC50 = 640 nM T89360 CMF8R1 22946293 IC50 = 43 nM T89360 CS42ZC 23626089 IC50 = 4100 nM T89360 CJO79M 23644735 Ki = 255 nM T89360 C2NW5X 23648220 Ki = 84 nM T89360 CCN63I 23648221 Ki = 143 nM T89360 CMVH63 23648222 Ki = 27 nM T89360 C0OR1M 23648223 Ki = 153 nM T89360 C5PIF4 23648224 Ki = 169 nM T89360 C90FQM 23648225 Ki = 49 nM T89360 CB35PV 23648226 Ki = 94 nM T89360 CQ90NK 23648227 Ki = 14 nM T89360 CKZT87 23648228 Ki = 108 nM T89360 CBC71W 23648229 Ki = 38 nM T89360 CH3Z4Q 24513583 IC50 > 5000 nM T89360 CBU17V 24513606 IC50 > 5000 nM T89360 CDXA20 24513641 IC50 > 5000 nM T89360 CZ8MT3 24517453 IC50 > 5000 nM T89360 CU94DR 24538043 IC50 > 5000 nM T89360 CYG18K 24748985 Ki = 540 nM T89360 C6M4QN 24748986 Ki = 1700 nM T89360 CK32AR 24749071 Ki = 1100 nM T89360 C9E0AU 24749072 Ki = 650 nM T89360 CG3O4V 24999500 IC50 > 5000 nM T89360 CO6DB0 25147739 Ki = 170 nM T89360 C09KIE 25181866 Ki = 1200 nM T89360 CND10S 25181867 Ki = 11000 nM T89360 CX5BU0 25181868 Ki = 340 nM T89360 C68PMG 25181869 Ki = 2600 nM T89360 C5JVN4 25210968 Ki = 8700 nM T89360 CUZT43 25210969 Ki = 2300 nM T89360 CW8I0P 25879063 IC50 = 87.7 nM T89360 CFU76P 26196040 IC50 = 1790 nM T89360 CS23HG 44024165 IC50 > 5000 nM T89360 C5IL9F 44024167 IC50 > 5000 nM T89360 C0F8KP 44275519 IC50 = 50 nM T89360 CQ2I6J 44275642 IC50 > 10000 nM T89360 C5YN8D 44275688 IC50 = 30 nM T89360 CQ4E9F 44275711 IC50 > 10000 nM T89360 CY8L1G 44275942 IC50 > 10000 nM T89360 CE0HC9 44276467 IC50 = 18 nM T89360 CEH64S 44276468 IC50 = 3800 nM T89360 C24IPY 44276469 IC50 = 740 nM T89360 C3DW1Z 44276622 IC50 = 550 nM T89360 C9YKC1 44276665 IC50 = 60 nM T89360 C4RZE0 44276698 IC50 = 820 nM T89360 CML9P3 44276709 IC50 = 3000 nM T89360 C1BZ8S 44276733 IC50 = 1660 nM T89360 C2BCQ0 44276734 IC50 = 740 nM T89360 CALV53 44276798 IC50 > 5000 nM T89360 CDB20G 44276803 IC50 > 5000 nM T89360 CZ2X8G 44276804 IC50 > 5000 nM T89360 C5GJ8H 44276818 IC50 > 1700 nM T89360 CD87HW 44276819 IC50 > 5000 nM T89360 CF18UY 44276869 IC50 = 150 nM T89360 C37KLD 44276961 IC50 = 400 nM T89360 C7TYB8 44276962 IC50 = 247 nM T89360 CT2Q0G 44276963 IC50 > 5000 nM T89360 CH3PF8 44277008 IC50 > 5000 nM T89360 CDS04H 44277009 IC50 = 1200 nM T89360 CIYN69 44304863 IC50 = 500 nM T89360 C0VD6L 44304866 IC50 > 5000 nM T89360 CS9FU7 44304883 IC50 = 41 nM T89360 CO3VX9 44304884 IC50 = 91 nM T89360 C50RLI 44304885 IC50 > 5000 nM T89360 CYF62T 44304900 IC50 > 5000 nM T89360 C84LXP 44304912 IC50 = 310 nM T89360 CH3UY4 44304932 IC50 = 100 nM T89360 CFG8V3 44305013 IC50 = 21 nM T89360 CSH83K 44305029 IC50 > 2000 nM T89360 CH6U5M 44305031 IC50 > 5000 nM T89360 CL60QO 44305034 IC50 > 1600 nM T89360 C0ZV6T 44305048 IC50 > 5000 nM T89360 C95JXK 44305067 IC50 = 1600 nM T89360 CNZ9E0 44305078 IC50 > 5000 nM T89360 CA3PV5 44305083 IC50 = 88 nM T89360 C94HVX 44305086 IC50 = 190 nM T89360 C7HFJ9 44305087 IC50 = 210 nM T89360 CNFR41 44305128 IC50 > 340 nM T89360 C27MSW 44305145 IC50 > 5000 nM T89360 CRQC38 44305148 IC50 > 57 nM T89360 CB40FT 44305192 IC50 > 5000 nM T89360 CKV9A4 44305213 IC50 > 2000 nM T89360 C7KEI3 44305214 IC50 > 2000 nM T89360 CGLZ25 44305233 IC50 > 5000 nM T89360 C5KRW0 44307938 IC50 = 72 nM T89360 CO0YU5 44308038 IC50 = 270 nM T89360 C3SEZ1 44308050 IC50 = 78 nM T89360 CGBD53 44308081 IC50 = 290 nM T89360 C2TN9P 44308105 IC50 = 3500 nM T89360 CAOH09 44308165 IC50 = 720 nM T89360 CYP86T 44308220 IC50 = 130 nM T89360 CKSV35 44308227 IC50 > 1000 nM T89360 CKSW94 44308417 IC50 = 250 nM T89360 CMP04J 44308425 IC50 = 620 nM T89360 CY2J8B 44329217 IC50 = 75 nM T89360 CLVU19 44329328 IC50 = 57 nM T89360 CQ1MW8 44329361 IC50 = 630 nM T89360 C2SG3Z 44329366 IC50 = 590 nM T89360 CRV1W0 44329410 IC50 > 3000 nM T89360 CFJ8S1 44329515 IC50 = 960 nM T89360 C7UX0J 44329529 IC50 = 110 nM T89360 C8GJN2 44329556 IC50 = 630 nM T89360 CA8P2J 44329800 IC50 > 1000 nM T89360 CPS1I4 44329801 IC50 = 2500 nM T89360 CMZ1T2 44329808 IC50 = 810 nM T89360 CF8P9E 44329815 IC50 > 1000 nM T89360 C50YRM 44330611 IC50 = 330 nM T89360 CZ2BR4 44330738 IC50 > 3000 nM T89360 C2N5CJ 44330750 IC50 = 130 nM T89360 CZ9UE0 44330773 IC50 = 340 nM T89360 CW8LY7 44330809 IC50 = 660 nM T89360 C07CSW 44330826 IC50 > 3000 nM T89360 CG17NB 44330827 IC50 = 240 nM T89360 CBN9J6 44330828 IC50 = 340 nM T89360 CB1VJ4 44336201 IC50 = 110 nM T89360 C4J8MO 44340409 IC50 = 40 nM T89360 C8BTY0 44340410 IC50 = 11 nM T89360 CL3OG8 44340423 IC50 = 200 nM T89360 C5FE6B 44340424 IC50 = 35 nM T89360 COW8S4 44340430 IC50 = 205 nM T89360 CQ4S0B 44340431 IC50 = 38 nM T89360 C9GB2W 44340450 IC50 > 5000 nM T89360 CLXS31 44340666 IC50 = 93 nM T89360 CU5N8R 44340674 IC50 > 5000 nM T89360 CX5HD2 44340724 IC50 = 35 nM T89360 CQC6A8 44340732 IC50 = 77 nM T89360 CRV2S9 44345136 IC50 = 84 nM T89360 CW4D9K 44345137 IC50 = 266 nM T89360 CHX1C3 44345138 IC50 = 6 nM T89360 CHJ67K 44345267 IC50 = 290 nM T89360 CQ52KT 44345310 IC50 = 420 nM T89360 C1AN9S 44345333 IC50 = 260 nM T89360 CTO57X 44354730 IC50 > 100000 nM T89360 CJ3N4G 44354906 IC50 = 89.8 nM T89360 CX9C7V 44355016 IC50 = 975 nM T89360 C4I3GD 44367217 IC50 = 160 nM T89360 CE9OC4 44367244 IC50 = 19 nM T89360 CB41DS 44367248 IC50 = 43 nM T89360 C5X1GF 44367255 IC50 = 46 nM T89360 C91HWG 44367420 IC50 = 26 nM T89360 CG45ZL 44367512 IC50 = 83 nM T89360 CU1VX2 44367513 IC50 < 10 nM T89360 C0RXO6 44367526 IC50 = 65 nM T89360 CXM9L0 44367538 IC50 = 5 nM T89360 CWIO57 44367546 IC50 = 180 nM T89360 CRE48F 44367552 IC50 = 65 nM T89360 CJR86I 44367578 IC50 = 29 nM T89360 CZID50 44367579 IC50 < 5 nM T89360 CY0OA1 44367590 IC50 > 10000 nM T89360 CZSP50 44367614 IC50 = 43 nM T89360 CZYC59 44367615 IC50 = 5 nM T89360 CY2J7R 44367639 IC50 = 30 nM T89360 CT5DZ1 44367690 IC50 = 21 nM T89360 COXS41 44367703 IC50 < 50 nM T89360 CS45OJ 44367718 IC50 = 33 nM T89360 CZU5N0 44367719 IC50 = 21 nM T89360 C4SOR5 44367730 IC50 = 5 nM T89360 C6VAS4 44367731 IC50 = 53 nM T89360 CM9S8K 44367733 IC50 = 140 nM T89360 CM06LV 44367743 IC50 = 15 nM T89360 CJ98VU 44367747 IC50 = 15 nM T89360 CR65TE 44390711 IC50 = 30 nM T89360 CSX2D6 44390718 IC50 = 17 nM T89360 C34JFM 44390721 IC50 = 91 nM T89360 CUY3T1 44390765 IC50 = 47 nM T89360 C1SNV9 44390777 IC50 = 22 nM T89360 CFI5P2 44390789 IC50 = 1710 nM T89360 CBQ8I7 44390790 IC50 = 100 nM T89360 C4P1JT 44390791 IC50 = 297 nM T89360 C8RDA1 44390811 IC50 = 821 nM T89360 C5B2FZ 44390828 IC50 = 71 nM T89360 CPZ9H5 44405422 IC50 = 192 nM T89360 C5LNB2 44405423 IC50 = 94 nM T89360 CN3O2U 44405428 IC50 = 49 nM T89360 C4FC9Y 44405429 IC50 = 328 nM T89360 CL0AE9 44405441 IC50 = 526 nM T89360 CNKD60 44405446 IC50 = 96 nM T89360 CK3PY1 44405447 IC50 = 104 nM T89360 C3R6PV 44405453 IC50 = 80 nM T89360 C7ZP0M 44405472 IC50 = 51 nM T89360 CZR84O 44405475 IC50 = 45 nM T89360 CY5N0I 44405476 IC50 = 68 nM T89360 CM0OF7 44405514 IC50 = 119 nM T89360 CH53NE 44405515 IC50 = 393 nM T89360 CR2Z7O 44405520 IC50 = 64 nM T89360 CG43TN 44405539 IC50 = 369 nM T89360 C5MA9V 44405578 IC50 = 71 nM T89360 CES5D6 44405580 IC50 = 79 nM T89360 CB43CW 44405581 IC50 = 948 nM T89360 CLG35S 44410469 IC50 = 71800 nM T89360 C3JM4T 44410476 IC50 = 222 nM T89360 CRP9B7 44410594 IC50 = 17000 nM T89360 CNE08X 44410595 IC50 = 1170 nM T89360 C0G5WM 44410601 IC50 = 128 nM T89360 C5R1BT 44410602 IC50 = 19500 nM T89360 C3SZT7 44410608 IC50 = 1360 nM T89360 COY6D8 44410643 IC50 = 4040 nM T89360 C8L3EA 44410644 IC50 = 7680 nM T89360 C6CS4Y 44410726 IC50 = 21000 nM T89360 C8ZP5U 44410728 IC50 = 7850 nM T89360 CO6K7B 44410732 IC50 = 58400 nM T89360 C8H4ES 44410734 IC50 = 6210 nM T89360 C48CJL 44410735 IC50 = 364 nM T89360 CJ81XI 44410872 IC50 = 27900 nM T89360 CMAZ04 44412558 IC50 = 246 nM T89360 CFQA81 44412573 IC50 > 1000 nM T89360 CL8JF5 44412582 IC50 = 273 nM T89360 C4PO0Y 44412597 IC50 = 96 nM T89360 CR61JY 44412598 IC50 = 86 nM T89360 CW4YP0 44412618 IC50 = 506 nM T89360 C4P8QV 44412632 IC50 = 68 nM T89360 C4Y6EC 44412633 IC50 = 24 nM T89360 CP0LU8 44412648 IC50 = 132 nM T89360 C1UP8I 44412712 IC50 = 93 nM T89360 C95XHE 44412713 IC50 > 1000 nM T89360 CFP3B7 44412731 IC50 > 1000 nM T89360 CR4N1Y 44412759 IC50 = 499 nM T89360 C5EP3N 44412773 IC50 = 785 nM T89360 C8LRG7 44412774 IC50 = 749 nM T89360 CAQC52 44412793 IC50 = 498 nM T89360 C70YFO 44415246 Ki = 60 nM T89360 CRZW96 44415248 Ki = 37 nM T89360 C16EMS 44433349 IC50 = 72000 nM T89360 CC2UO4 44440695 IC50 = 18800 nM T89360 CY6SQ1 44458844 IC50 = 150 nM T89360 C0RU5A 44458846 IC50 = 290 nM T89360 C14SVM 44458898 IC50 > 1000 nM T89360 COQ83H 44578784 IC50 = 18800 nM T89360 C84EYU 44578785 Ki = 310 nM T89360 C8GJB9 44578786 Ki = 180 nM T89360 C9T2EI 44578787 Ki = 440 nM T89360 CIK76G 44578789 Ki > 100000 nM T89360 CEI32X 44589747 Ki = 14300 nM T89360 C2MF0S 44589785 Ki > 100000 nM T89360 CG7WJ4 44589786 Ki = 30100 nM T89360 C7Y9QT 44602364 IC50 > 5000 nM T89360 CM2U4H 45257259 IC50 > 5000 nM T89360 CAH41O 45257352 IC50 > 5000 nM T89360 C7OGF2 45257354 IC50 > 5000 nM T89360 CVO20H 46839190 Ki = 2200 nM T89360 C3GET9 46839191 Ki = 34 nM T89360 C0SV8O 46839192 Ki = 200 nM T89360 C1V3CQ 46839320 Ki = 44 nM T89360 CH6S4E 46871958 IC50 > 5000 nM T89360 CG2JO0 46876259 Ki = 300 nM T89360 C01DSF 46876831 Ki = 950 nM T89360 CG3RM9 46876832 Ki = 290 nM T89360 CJQ8D6 46898106 IC50 > 5000 nM T89360 CIT31Y 46927861 Ki = 250 nM T89360 CXW02B 46927862 Ki = 120 nM T89360 CU4Z3R 49864088 Ki = 1400 nM T89360 CP5HR1 49864089 Ki = 1500 nM T89360 CQ39WM 49864090 Ki = 230 nM T89360 C76JYP 49864102 Ki = 1200 nM T89360 CN2G3Z 49864103 Ki = 1800 nM T89360 C01GAC 49864104 Ki = 200 nM T89360 CR8E0Z 51351534 Ki = 24 nM T89360 C9YL2W 51351535 Ki = 73 nM T89360 CPY1M0 51351558 Ki = 38 nM T89360 C09MCD 52589406 IC50 > 5000 nM T89360 CT64YQ 52905544 Ki = 487 nM T89360 C81NCO 53317433 Ki = 770 nM T89360 C81TOB 53317434 Ki = 167 nM T89360 C7R4DT 53317435 Ki = 83 nM T89360 CZ4FR9 53317436 Ki = 34 nM T89360 C0MC6P 53320028 Ki = 3770 nM T89360 C64FAH 53320029 Ki = 6600 nM T89360 CQU37F 53320030 Ki = 39 nM T89360 CFO5E7 53320031 Ki = 44 nM T89360 CN32LO 53320311 Ki = 84 nM T89360 CPO0F3 53322659 Ki = 60 nM T89360 CMT39Y 53322660 Ki = 1900 nM T89360 CN6Q8M 53324226 Ki = 14 nM T89360 CC9D8J 53326788 Ki = 30 nM T89360 C6HQ7S 56835081 IC50 = 2100 nM T89360 C18UZI 56835082 IC50 = 4500 nM T89360 C91ARE 56835083 IC50 = 8800 nM T89360 CNGX19 56835085 IC50 = 3200 nM T89360 C5HZ3Q 56835102 IC50 = 2800 nM T89360 CP32QL 57391310 IC50 > 5000 nM T89360 CBMX91 57391311 IC50 > 5000 nM T89360 CCZ98A 57393086 IC50 > 5000 nM T89360 CK1RZ4 57394813 IC50 > 5000 nM T89360 C5BNH7 57396578 IC50 > 5000 nM T89360 C3HKO1 57398354 IC50 > 5000 nM T89360 CMAT05 57398355 IC50 > 5000 nM T89360 CM7T2I 57398356 IC50 > 5000 nM T89360 C6V0XL 57398357 IC50 > 5000 nM T89360 C3XD9L 57400014 IC50 > 5000 nM T89360 CR6AE3 57400851 IC50 = 400 nM T89360 C7HF5T 57401823 IC50 > 5000 nM T89360 C4IE8C 57401824 IC50 > 5000 nM T89360 CY5L8X 57401825 IC50 > 5000 nM T89360 CF79PO 57403530 IC50 > 5000 nM T89360 CC54BA 57403531 IC50 > 5000 nM T89360 C09ZCY 59053796 IC50 = 28860 nM T89360 C48TLR 59053798 IC50 = 73240 nM T89360 CB9G6K 67473072 IC50 >= 5000 nM T89360 C4DG7M 67473106 IC50 > 5000 nM T89360 CHW41M 67473122 IC50 >= 5000 nM T89360 C87ORP 67473132 IC50 >= 5000 nM T89360 CEU7I8 67473135 IC50 >= 5000 nM T89360 C3WLG5 67473139 IC50 >= 5000 nM T89360 CO5U4S 70693788 IC50 = 6430 nM T89360 C3IQE9 70850880 IC50 > 5000 nM T89360 CH26JV 70851038 IC50 > 5000 nM T89360 CF53JE 71297189 IC50 > 5000 nM T89360 CFA3N8 71450059 IC50 >= 5000 nM T89360 CMI97N 71453700 IC50 >= 5000 nM T89360 CW3VL9 71453701 IC50 >= 5000 nM T89360 CM05XU 71455424 IC50 >= 5000 nM T89360 C61ATW 71455425 IC50 >= 5000 nM T89360 C3AT8D 71462576 IC50 >= 5000 nM T89360 CZAV85 71462577 IC50 >= 5000 nM T89360 CMVL76 71661540 IC50 > 5000 nM T89360 C1V5AQ 71661543 IC50 > 5000 nM T89360 CX5WE1 71661544 IC50 > 5000 nM T89360 CV1D5W 71661721 IC50 > 5000 nM T89360 CNIJ92 71661722 IC50 > 5000 nM T89360 CO36TX 71661724 IC50 > 5000 nM T89360 CZ1TF2 71661725 IC50 > 5000 nM T89360 CW54QI 71661894 Ki > 5000 nM T89360 CC9U7A 71661895 IC50 > 5000 nM T89360 C8CX0T 71661896 IC50 > 5000 nM T89360 C6RN9G 71661897 IC50 > 5000 nM T89360 CI6YS9 71662079 IC50 > 5000 nM T89360 C87LXA 71662080 IC50 > 5000 nM T89360 C51OLK 71662081 Ki > 5000 nM T89360 C2ILR9 71662082 IC50 > 5000 nM T89360 C7IQA2 71662258 IC50 > 5000 nM T89360 CD35JI 71662259 IC50 > 5000 nM T89360 CIFH53 71662260 IC50 > 5000 nM T89360 CRB19S 71662261 IC50 > 5000 nM T89360 CP6WC3 71662422 IC50 > 5000 nM T89360 C6T5XE 71662423 IC50 > 5000 nM T89360 CE0ON2 71662424 IC50 > 5000 nM T89360 CD9UX5 71662426 IC50 > 5000 nM T89360 CYT20K 71662586 IC50 > 5000 nM T89360 CO8V4B 71662587 IC50 > 5000 nM T89360 CC0A9E 71662588 IC50 > 5000 nM T89360 C50TWZ 71662589 IC50 > 5000 nM T89360 C9GAL6 71662590 IC50 > 5000 nM T89360 CX58GA 71662775 Ki > 5000 nM T89360 C8N7CG 71662776 IC50 > 5000 nM T89360 CC3WB6 71662779 IC50 > 5000 nM T89360 CDVK12 71662780 IC50 > 5000 nM T89360 C39KQY 71716568 IC50 = 90 nM T89360 C3M0JK 72163956 IC50 = 98 nM T89360 CNQ2D6 72945146 Ki = 165 nM T89360 C5OJ0X 72945148 Ki = 186 nM T89360 C01HVL 72945149 Ki = 102 nM T89360 C1OVC0 72945150 Ki = 231 nM T89360 CBPC50 72945349 Ki = 84 nM T89360 C7MJQ5 72945350 Ki = 967 nM T89360 C9NTH1 72945351 Ki = 175 nM T89360 CVJ0N8 72945352 Ki = 70 nM T89360 CP1I9N 72945353 Ki = 1964 nM T89360 CJ4R8C 72945541 Ki = 1227 nM T89360 C74WCI 72945542 Ki = 88 nM T89360 C7T3HN 72945732 Ki = 24 nM T89360 C95BZQ 72947911 Ki = 15 nM T89360 CCVO01 72947912 Ki = 14 nM T89360 CB7HG8 72948102 Ki = 37 nM T89360 C4U3OA 72948103 Ki = 56 nM T89360 CX2U3L 72948104 Ki = 44 nM T89360 C3N7OD 72948105 Ki = 749 nM T89360 CZJ5F6 73346517 Ki = 2398 nM T89360 CN5QE0 73346518 Ki = 321 nM T89360 C26EXZ 73349141 IC50 = 330 nM T89360 CAD90T 73349545 Ki = 437 nM T89360 CD4BY1 73351103 Ki = 2672 nM T89360 CB94EM 73352218 IC50 = 387 nM T89360 CWO9Q0 73352572 Ki = 163 nM T89360 CPS4I8 76309998 Ki = 12.6 nM T89360 CB2PT6 76309999 Ki = 40 nM T89360 CL42ER 76310000 Ki = 215 nM T89360 CI1J4W 76310001 Ki = 94 nM T89360 CEB47C 76310002 Ki = 2790 nM T89360 C3ICR7 76310003 Ki = 524 nM T89360 C7C9FJ 76317234 Ki = 235 nM T89360 CTLJ38 76317235 Ki = 364 nM T89360 CZ9U2T 76320941 Ki = 233 nM T89360 C7HJC1 76324606 Ki = 188 nM T89360 C0DFQ1 76328163 Ki = 438 nM T89360 CL41TU 76328164 Ki = 134 nM T89360 C86TRQ 76331843 Ki = 174 nM T89360 CTFG08 76331844 Ki = 147 nM T89360 C3OVW6 76335415 Ki = 188 nM T89360 CG7Z4S 76335416 Ki = 188 nM T89360 C72ZFE 90663687 IC50 = 800 nM T89360 CD9S8B 90663694 Ki = 110 nM T89360 CC6RG7 90663712 IC50 = 175000 nM T89360 CEX1D3 90663714 IC50 = 800 nM T89360 C0A3ZW 90663715 IC50 = 6000 nM T89360 C47LAF 135418940 IC50 > 10000 nM T89360 CJVW76 135419254 IC50 = 52800 nM T89360 C8J2PC 135456762 IC50 > 10000 nM T89360 CEDB45 135500033 IC50 = 18 nM T89360 C4BFY3 135566969 IC50 > 10000 nM T89360 C0USX4 135883678 IC50 = 740 nM T89360 CM9QB3 135883679 IC50 = 800 nM T89360 C3GW8I 135883680 IC50 > 1000 nM T89360 CIT3E5 135976449 IC50 = 37000 nM T89360 C25EPJ 135976460 IC50 > 1000000 nM T89360 CMG6I4 135976469 IC50 = 440 nM T89360 CV4G0A 135976470 IC50 > 1000000 nM T89360 CQ4T2N 135976471 IC50 = 132000 nM T89360 CF0GR8 135976472 IC50 > 1000000 nM T89360 CTZ82I 135976473 IC50 = 1200 nM T89360 CV9WK5 135976474 IC50 = 1000 nM T89360 C5W3TV 135976476 IC50 = 1320 nM T89360 C0UR9J 135976481 IC50 = 460000 nM T89360 CTF7A4 136042356 IC50 > 5000 nM T89360 CY94ZB 136215772 IC50 > 10000 nM T89360 C7JEG1 136215773 IC50 > 10000 nM T89360 CF7O2U 136215774 IC50 > 10000 nM T89360 CFP0V5 136215897 IC50 > 10000 nM T89360 C3NHA6 136219159 IC50 > 5000 nM T89360 CG75EV 138393087 Ki > 5000 nM T89360 C1GPY5 145952889 IC50 = 1500 nM T89360 CFQ2O9 145954131 IC50 > 30000 nM T89360 C8O2IJ 145963797 Ki > 5000 nM T89360 C40WKT 145964095 Ki > 5000 nM T89360 CR78JK 145964212 Ki > 5000 nM T89360 CFS5Z3 145964258 Ki > 5000 nM T89360 CC3T5V 145964499 Ki > 5000 nM T89360 C0KGT4 145964791 Ki > 5000 nM T89360 CJAI17 145964939 Ki > 5000 nM T89360 C3AXP6 145965235 Ki > 5000 nM T89360 CW50CM 145965999 Ki > 5000 nM T89360 CB4NX2 145966576 Ki > 5000 nM T89360 C5V7ZK 145966629 Ki > 5000 nM T89360 C8E7TL 145966683 Ki > 5000 nM T89360 C02DKL 145966779 Ki > 5000 nM T89360 C5K3DS 145967011 Ki > 5000 nM T89360 C1AD8R 145967013 Ki > 5000 nM T89360 CYTB64 145967134 Ki > 5000 nM T89360 C9EZ5L 145970298 Ki > 5000 nM T89360 C4RNH8 145970986 Ki = 2900 nM T89360 C5GW7N 145971015 Ki > 5000 nM T89360 CA6C2F 145972082 Ki > 5000 nM T89360 C2PV6E 145972358 Ki > 5000 nM T89360 CTV68U 145972501 Ki > 5000 nM T89360 C5HCJ8 145972590 Ki > 5000 nM T89360 CI31YE 145972757 IC50 = 4540 nM T89360 CFS82G 145973482 Ki > 5000 nM T89360 C06FRK 145974169 Ki > 5000 nM T89360 C1KSO5 145974525 Ki = 3300 nM T89360 C8B7LI 145974642 Ki > 5000 nM T89360 C24ZLQ 145974896 Ki > 5000 nM T89360 C1VID9 145975055 Ki > 5000 nM T89360 C7RUP4 145975474 Ki > 5000 nM T89360 C23DWC 145975793 Ki > 5000 nM T89360 CR1ND4 145975885 Ki > 5000 nM T89360 C3ZQ7I 145976477 Ki = 2000 nM T89360 C48WSM 145976500 Ki > 5000 nM T89360 CHA9M2 145976564 Ki > 5000 nM T89360 C1KJ4W 145977312 Ki > 5000 nM T89360 CC1L4J 145977399 Ki > 5000 nM T89360 C2GU3O 145977423 Ki > 5000 nM T89360 CG86KY 145977474 Ki > 5000 nM T89360 CTGB02 145977680 Ki > 5000 nM T89360 CJX17G 145977828 Ki = 2300 nM T89360 CZK4L8 145978048 Ki > 5000 nM T89360 CQF9Z2 145978149 Ki > 5000 nM T89360 C06RKZ 145978312 Ki > 5000 nM T89360 C24OSG 145979776 IC50 = 7380 nM T89360 C93AKF 145980356 IC50 = 1600 nM T89360 C67YXK 145980711 IC50 = 4200 nM T89360 CUSP05 145981621 IC50 = 360 nM T89360 C10YDI 145982128 IC50 = 430 nM T89360 CWC78S 145983656 IC50 = 1200 nM T89360 C6VP2S 145985880 IC50 > 30000 nM T89360 CPLR18 145988080 IC50 = 570 nM T89360 C1K4BC 145989436 IC50 = 360 nM T89360 C5QBJ2 145989469 IC50 = 4400 nM T89360 CCY78M 145990077 IC50 = 660 nM T89360 C20PUW 145990385 IC50 = 2200 nM T89360 CIG96S 145990435 IC50 = 790 nM T89360 CBL59V 145990969 IC50 = 4500 nM T89360 CP42FJ 145991406 IC50 = 1200 nM T89360 D01LDQ 24749070 Ki = 30 nM T89360 D02YMQ 44410733 IC50 = 456 nM T89360 D03HDS 6475540 Ki = 380 nM T89360 D04LRN 22238481 IC50 = 600 nM T89360 D05SKE 44410796 IC50 = 408 nM T89360 D06FSR 2307681 IC50 = 7660 nM T89360 D06RQV 44410708 IC50 = 419 nM T89360 D07BPT 135457978 IC50 > 10000 nM T89360 D07HZQ 444451 Ki = 21 nM T89360 D08OSM 10607518 IC50 = 5840 nM T89360 D0A0UW 22238483 IC50 = 500 nM T89360 D0A4AL 477579 Ki = 250 nM T89360 D0AL2E 44410707 IC50 = 524 nM T89360 D0B2WX 135407310 IC50 > 10000 nM T89360 D0D1KZ 87894 IC50 = 6840 nM T89360 D0D2ST 11962095 IC50 = 343 nM T89360 D0E5EW 135531482 IC50 > 10000 nM T89360 D0G3BY 44410465 IC50 = 15400 nM T89360 D0GA0Y 135463623 IC50 > 10000 nM T89360 D0H1II 510913 IC50 = 630 nM T89360 D0J9OS 44410800 IC50 = 6210 nM T89360 D0K4EM 44410928 IC50 = 637 nM T89360 D0L0MJ 644354 IC50 = 1150 nM T89360 D0L0ZP 15462732 IC50 = 8200 nM T89360 D0Q3WC 44410473 IC50 = 1110 nM T89360 D0S4BK 73680 Ki = 100 nM T89360 D0T4UE 44578788 Ki = 4000 nM T89360 D0V0YP 44410875 IC50 = 2320 nM T89360 D0Y1MH 135471354 IC50 > 10000 nM T89360 D0Z0YB 16748635 IC50 = 2200 nM T89360 D0Z8EV 446541 Ki = 6 nM T89360 D0ZG3O 44410730 IC50 = 586 nM T08741 D0E6XR 3062316 IC50 = 1.3 nM T08741 D0EG1I 9926791 IC50 > 10000 nM T08741 D0OB0F 5328940 IC50 = 63 nM T08741 D02UFQ 11620908 IC50 = 4700 nM T08741 D03LWG 53235510 IC50 > 10000 nM T08741 D04AHQ 71721540 IC50 = 290 nM T08741 D07EHV 44814409 IC50 > 10000 nM T08741 D07HPJ 11476171 IC50 > 10000 nM T08741 D0E3TC 44259 IC50 = 14.3 nM T08741 D0M0XB 10302451 IC50 = 840 nM T08741 D0Q7RE 16007391 Ki > 10000 nM T08741 D0VF6E 1401 IC50 = 19800 nM T08741 D03BNU 59604787 IC50 > 10000 nM T08741 D09HEV 6539952 IC50 = 41 nM T08741 D0T3ME 156422 IC50 > 30000 nM T08741 CB1VW3 1400 IC50 = 640 nM T08741 CJ17AM 4877 IC50 = 1970 nM T08741 C7E5WO 72779 IC50 = 75000 nM T08741 CWGJ94 256524 IC50 = 9500 nM T08741 C5RK3H 5330188 IC50 = 7300 nM T08741 CD7U5B 5330196 IC50 = 2000 nM T08741 CB23PA 5330197 IC50 = 1700 nM T08741 CPXK25 5793057 IC50 = 6850 nM T08741 CB7WK3 5938113 IC50 > 100000 nM T08741 CP0XI6 6603792 IC50 = 5180 nM T08741 CR2B8U 9888491 IC50 > 10000 nM T08741 CG6A1H 9927800 IC50 > 10000 nM T08741 CJO47T 9948405 IC50 > 10000 nM T08741 CV8I5X 9999342 IC50 > 10000 nM T08741 C5TQ7X 10247543 IC50 > 10000 nM T08741 C8RD3V 10301884 IC50 = 270 nM T08741 CFLH53 10432113 IC50 > 5000 nM T08741 CL7PF2 10451087 IC50 = 5000 nM T08741 C2WQ8M 10473563 IC50 > 10000 nM T08741 CACS26 11561968 Ki > 2000 nM T08741 CSM62L 11626920 IC50 > 30000 nM T08741 CU0E8O 11690457 Ki > 2000 nM T08741 CZY05V 11719421 IC50 = 659 nM T08741 C1OK2P 14147704 IC50 = 15500 nM T08741 CQ9Z0L 15550318 IC50 > 10000 nM T08741 CP8OW6 15858662 IC50 > 5000 nM T08741 C9TU1O 16046126 IC50 > 1000 nM T08741 CL0XQ4 16094815 IC50 = 47000 nM T08741 CBM09R 16094816 IC50 = 21000 nM T08741 CKG9E6 16094817 IC50 = 34000 nM T08741 C4I1GM 16094818 IC50 = 3300 nM T08741 CRH81B 16094819 IC50 = 4900 nM T08741 CQ25BA 16094820 IC50 = 11000 nM T08741 C20YKV 16094821 IC50 = 18000 nM T08741 C5SAU7 16094822 IC50 = 5600 nM T08741 C39GBM 16094823 IC50 = 3400 nM T08741 CS0E2L 16094824 IC50 = 57000 nM T08741 CG35DT 16094827 IC50 = 29000 nM T08741 CN4F5Q 16094828 IC50 = 290000 nM T08741 CSAD50 16094829 IC50 = 2500 nM T08741 C6BQE5 16094830 IC50 = 291000 nM T08741 CH4D6T 16094831 IC50 = 28000 nM T08741 CN03HF 16094832 IC50 = 7000 nM T08741 CT7AK0 16094834 IC50 = 12000 nM T08741 CZ2D6G 16094835 IC50 = 6100 nM T08741 C0EF7G 16094836 IC50 = 6300 nM T08741 CB6YP5 16094837 IC50 = 3200 nM T08741 CWF48O 16094838 IC50 = 3400 nM T08741 CQL45G 16094839 IC50 = 18000 nM T08741 CQG45C 16109001 IC50 = 25000 nM T08741 C1U8XW 16109036 IC50 = 1800 nM T08741 C0E2OG 20579089 IC50 > 10000 nM T08741 CG6D4M 23647319 IC50 > 10000 nM T08741 CY8Z7X 23647330 IC50 > 10000 nM T08741 C4XD8H 23647348 IC50 > 10000 nM T08741 CQNP54 24764449 IC50 = 165 nM T08741 C0P6AU 24894017 IC50 = 80 nM T08741 CBK82P 25011729 IC50 = 10700 nM T08741 CEL61X 44229839 IC50 = 3900 nM T08741 C1KSW5 44335197 IC50 > 5000 nM T08741 CV0F4D 44384547 IC50 > 5000 nM T08741 CI2L9R 44384964 IC50 > 5000 nM T08741 CC09FT 44384965 IC50 = 4300 nM T08741 CV8LS1 44418760 IC50 = 9500 nM T08741 C3VRO9 44557921 IC50 > 10000 nM T08741 C1J6GR 46224908 IC50 = 4.5 nM T08741 CHSF07 49806372 IC50 > 1000 nM T08741 CEQN27 52936621 Ki > 1000 nM T08741 C8NA4L 53384644 IC50 > 30000 nM T08741 CJ47MX 56963907 IC50 = 10000 nM T08741 C9L6FD 56963908 IC50 > 10000 nM T08741 CE50IB 56963909 IC50 > 10000 nM T08741 CT3EW2 59292007 IC50 > 1000 nM T08741 C1MR8Q 60097495 IC50 > 10000 nM T08741 CV63UL 67240318 IC50 > 10000 nM T08741 C8I7GC 68293638 IC50 > 10000 nM T08741 C82FIP 70686752 IC50 = 3100 nM T08741 C0QX3Y 70688829 IC50 = 2600 nM T08741 CSOT12 70693058 IC50 > 10000 nM T08741 CS6NW3 70693059 IC50 = 10000 nM T08741 COU73Y 71226944 IC50 = 261 nM T08741 C40JOZ 71235465 IC50 = 626 nM T08741 CEBO91 71452977 IC50 = 5100 nM T08741 CZ31PU 71583657 IC50 > 10000 nM T08741 C2AN7T 134611886 IC50 > 100000 nM T08741 CZFA70 135611366 IC50 = 704 nM T08741 CYDM01 135891431 IC50 = 1.7 nM T08741 CZOD53 137633880 IC50 = 1154 nM T08741 C7BJY5 137636807 IC50 = 665 nM T08741 CO89DX 137649100 IC50 = 455 nM T08741 CINE03 137652514 IC50 = 2145 nM T08741 C28QUP 137652864 IC50 = 2826 nM T08741 CLJH31 139209093 IC50 = 42 nM T08741 CVI30A 139600340 IC50 < 3 nM T08741 C6VB3O 145925651 IC50 >= 5000 nM T08741 CF27EG 155511610 IC50 = 402 nM T08741 C0AN1O 155512752 IC50 = 473 nM T08741 C8TL1A 155513050 IC50 = 8 nM T08741 C2MD1Q 155513187 IC50 > 10000 nM T08741 CEDI24 155516854 IC50 = 4 nM T08741 C3V4LG 155538413 IC50 = 706 nM T08741 CGDJ81 155539793 IC50 = 21 nM T08741 CDW9G6 155541623 IC50 = 80 nM T08741 CLJ80U 155548662 IC50 = 4 nM T08741 CGTR28 155552797 IC50 < 3 nM T08741 CCV06Q 155554126 IC50 < 3 nM T08741 C3DQI8 155557074 IC50 = 79 nM T08741 CVS68Y 155558083 IC50 = 5600 nM T08741 CT8VX1 155562023 IC50 < 3 nM T08741 CR6EL3 155568078 IC50 = 430 nM T08741 C12HQW 155568509 IC50 = 70 nM T08741 D06HVH 54613583 IC50 > 10000 nM T08741 D06LJL 9916282 IC50 = 21000 nM T08741 D0BU6T 354471 IC50 > 5000 nM T08741 D0GT8N 5154691 IC50 = 510 nM T08741 D0IR6U 5494425 IC50 = 2100 nM T08741 D0L4WN 31420 IC50 > 40000 nM T08741 D0P6JS 11675054 IC50 > 10000 nM T89039 D01ZSO 4235 Ki > 200 nM T89039 D0D1AL 3559 Ki = 16 nM T89039 D0H2SE 118607347 Ki = 48 nM T89039 D0W3TS 41306362 Ki = 190 nM T89039 D0XK2K 9829526 Ki = 0.12 nM T89039 C7B8VJ 44405080 Ki = 1550 nM T89039 CLY10I 65659 Ki > 200 nM T89039 CI8KD2 97627 Ki = 796 nM T89039 CS4XQ9 1081502 Ki > 200 nM T89039 C6Z4QI 3050372 Ki = 25.1 nM T89039 C5NA6S 3069135 Ki = 5.12 nM T89039 C6AX8Y 3126148 Ki > 200 nM T89039 C4Z0DT 9049339 Ki = 160 nM T89039 CTAC24 9885114 Ki = 231 nM T89039 CZ9MG4 10356384 Ki > 200 nM T89039 C5F4WP 10403711 Ki = 4350 nM T89039 CC1AT3 11165837 Ki = 10.33 nM T89039 CBFZ60 11531451 Ki = 113 nM T89039 C1HDM5 11653679 Ki = 5.129 nM T89039 CCG14E 13091356 Ki = 18 nM T89039 CYN95Z 13091359 Ki = 29 nM T89039 C65SCN 15599151 Ki = 432 nM T89039 CTME96 16202156 Ki = 0.26 nM T89039 C45JHX 17644936 Ki > 200 nM T89039 C7MST8 17758676 Ki = 12.6 nM T89039 CCM1L3 18118650 Ki = 340 nM T89039 CZ31UL 18118651 Ki > 1200 nM T89039 C9UE6C 18118654 Ki > 1200 nM T89039 CWQ5S7 27148262 Ki = 360 nM T89039 C4MRQ0 27842480 Ki = 2750 nM T89039 CUVS17 29048070 Ki = 95 nM T89039 C7EJK2 31588412 Ki = 321 nM T89039 CO9HV7 40624141 Ki > 1200 nM T89039 CRJ5E1 41306333 Ki > 1200 nM T89039 CCF93H 41306385 Ki = 350 nM T89039 CQSO71 41306434 Ki > 1200 nM T89039 CGO25K 41306445 Ki = 310 nM T89039 C83TBP 41307231 Ki = 200 nM T89039 CK5Z6Q 45160790 Ki = 1995.26 nM T89039 C3A9OY 51111240 Ki = 470 nM T89039 CPJZ31 52149645 Ki = 200 nM T89039 C82HKM 52750322 Ki = 160 nM T89039 CIW0F6 54582640 Ki = 227 nM T89039 CZU6L2 57345618 Ki = 5.888 nM T89039 CK9G8H 57345619 Ki = 8.5 nM T89039 C4EXS6 57396571 Ki = 33 nM T89039 CYN38R 57401819 Ki = 51.5 nM T89039 C3TNQ5 60346448 Ki = 850 nM T89039 C7JG9R 60701380 Ki > 400 nM T89039 C7FMA4 70676458 Ki = 2010 nM T89039 C28RIZ 76518514 Ki = 25.12 nM T89039 CLM0J5 90644067 Ki = 600 nM T89039 CH5R8Q 98049507 Ki = 32 nM T89039 CO6Z7J 110440208 Ki = 200 nM T89039 CBW0U9 110445832 Ki = 98 nM T89039 CHU07G 118607283 Ki = 170 nM T89039 CX2QI6 118607309 Ki = 1400 nM T89039 CIW02L 118607351 Ki = 200 nM T89039 C84QJX 118607364 Ki = 59 nM T89039 CX5B2A 118607439 Ki = 170 nM T89039 CXOT38 118607453 Ki = 49 nM T89039 C4U2GB 118607455 Ki = 20 nM T89039 CSB25E 118709750 Ki = 8.1 nM T89039 CD4S9R 118709751 Ki = 2.138 nM T89039 CM57GR 126720252 Ki = 1200 nM T89039 CN91JP 137632351 Ki = 8.4 nM T89039 CUV20T 137636134 Ki = 76.1 nM T89039 C4PAF3 137642542 Ki = 22.3 nM T89039 C5NL4A 137645149 Ki = 23 nM T89039 C92HOT 137650821 Ki = 23.8 nM T89039 C6GZR2 137653169 Ki = 24 nM T89039 CM7IN4 137657904 Ki = 16.2 nM T89039 CZG4P7 137662176 Ki = 25.5 nM T89039 C1TQ2A 145953153 Ki = 110 nM T89039 CXEV63 145954849 Ki = 5.19 nM T89039 CDGA65 145956728 Ki = 350 nM T89039 CJA9T4 146597626 Ki > 10000 nM T89039 C3D4UM 146597628 Ki > 10000 nM T89039 C7UHR0 146597630 Ki = 251.19 nM T89039 CCRS21 146597638 Ki > 10000 nM T89039 CM18OU 146597639 Ki = 630.96 nM T89039 C42TIZ 146597651 Ki = 398.11 nM T89039 CL5PG8 146597666 Ki > 10000 nM T89039 C89YUC 146597677 Ki > 10000 nM T89039 CU9G0O 146597678 Ki > 10000 nM T89039 C6TRC9 146641556 Ki > 10000 nM T89039 C8I3YJ 146641558 Ki = 100 nM T89039 C3LBA0 146641564 Ki > 10000 nM T89039 CFD4N9 146641568 Ki = 501.19 nM T89039 CP70WA 146641787 Ki > 10000 nM T89039 C0WU5Y 146641788 Ki > 10000 nM T89039 C10LOP 146641795 Ki = 251.19 nM T89039 CG97ER 146709966 Ki = 316.23 nM T89039 C6FX4M 147636204 Ki = 1000 nM T89039 CW4S2X 147652368 Ki > 10000 nM T89039 CF5B2L 147653864 Ki = 630.96 nM T89039 C5PNX8 148302367 Ki = 316.23 nM T89039 C2E5HK 149396365 Ki = 100 nM T89039 C9T0PS 153061504 Ki = 1995.26 nM T89039 CF7J3M 153287535 Ki = 3981.07 nM T89039 C72MVW 153287537 Ki = 1258.93 nM T89039 CAF36V 153287539 Ki = 79.43 nM T89039 C1FA0K 153287541 Ki = 316.23 nM T89039 CEQ69Z 153287542 Ki = 125.89 nM T89039 C9A7SV 153287550 Ki > 10000 nM T89039 C91KST 153287551 Ki = 1258.93 nM T89039 C6P3SR 153287553 Ki = 1000 nM T89039 C3G5CJ 153287557 Ki = 79.43 nM T89039 CW31CT 153287566 Ki = 158.49 nM T89039 CYP86E 153287567 Ki = 316.23 nM T89039 CS73ZC 153287568 Ki = 316.23 nM T89039 CV9G7Z 153287572 Ki > 10000 nM T89039 CO85KL 153287574 Ki = 630.96 nM T89039 CCD9N1 155512086 Ki = 753 nM T89039 CTV8R1 155512151 Ki = 642 nM T89039 CV35ZN 155513505 Ki = 662 nM T89039 C2D8ZF 155515129 Ki = 7.61 nM T89039 C58EAT 155515524 Ki = 11 nM T89039 C5K2GQ 155516317 Ki = 14 nM T89039 C4KWA1 155518665 Ki = 2.512 nM T89039 CUSA24 155519891 Ki > 10000 nM T89039 CU8D3T 155519913 Ki = 16 nM T89039 CIP3X7 155523942 Ki = 21.8 nM T89039 CY17EB 155524132 Ki = 4.6 nM T89039 CY5Q0J 155524744 Ki = 11 nM T89039 C9W2NV 155525645 Ki = 158.49 nM T89039 CP76JX 155526977 Ki > 10000 nM T89039 CW6CX1 155528147 Ki = 1673 nM T89039 CPA51T 155528865 Ki = 42.66 nM T89039 C3Z5XG 155529711 Ki = 7.6 nM T89039 C8RGT9 155532745 Ki = 5.5 nM T89039 CV83SG 155534733 Ki = 1720 nM T89039 C7PO3B 155535411 Ki = 64.1 nM T89039 C7PW0N 155535978 Ki = 8 nM T89039 CB79ZW 155536080 Ki > 10000 nM T89039 CIUS98 155536619 Ki = 2090 nM T89039 CR16NT 155540848 Ki = 39.81 nM T89039 CW76ES 155542765 Ki = 87 nM T89039 CMT60C 155543832 Ki = 349 nM T89039 CIA1C9 155547197 Ki = 32 nM T89039 CJ1U4N 155547337 Ki = 16 nM T89039 CF7MQ8 155550094 Ki > 10000 nM T89039 CI41QF 155552117 Ki = 2550 nM T89039 CJ92EA 155552895 Ki = 316.23 nM T89039 CKSZ39 155553997 Ki = 13 nM T89039 C04OFL 155554079 Ki = 2.2 nM T89039 CRU26E 155554287 Ki = 125.89 nM T89039 CZ9U5N 155554849 Ki = 251.19 nM T89039 C5EVM7 155555743 Ki = 651.6 nM T89039 CC48RQ 155556295 Ki = 25.12 nM T89039 CBS89O 155556618 Ki = 1170 nM T89039 CJBX01 155557042 Ki = 3162.28 nM T89039 C8TO2W 155558029 Ki = 1300 nM T89039 C4QID8 155558857 Ki = 6.7 nM T89039 CK4Z6D 155559218 Ki = 7.9 nM T89039 C4J0ZI 155559223 Ki > 10000 nM T89039 C13RCK 155561279 Ki = 13.1 nM T89039 CXYQ73 155561471 Ki = 31.62 nM T89039 CCOD50 155562467 Ki = 1980 nM T89039 C4N9GU 155563428 Ki = 2020 nM T89039 CK9RN6 155563452 Ki = 8.4 nM T89039 CSM7V1 155564110 Ki = 7.943 nM T89039 CR0F6E 155565622 Ki = 68.8 nM T89039 CBI7N3 155566272 Ki = 583 nM T89039 CNCT72 155568142 Ki = 3.8 nM T89039 C5N2EK 155568367 Ki > 1000 nM T89039 D02WJT 7333 Ki = 20 nM T89039 D0F0IA 11301655 Ki > 2000 nM T89039 D0KL1P 10474335 Ki = 0.34 nM T89039 D0P0XA 197060 Ki = 90.4 nM T89039 D0Q7FM 15443 Ki = 50.12 nM T55293 CU8E4T 16657205 IC50 = 50000 nM T55293 CZDU14 45268344 IC50 = 2380 nM T55293 CZY12B 45270076 IC50 > 100000 nM T16347 D03DXN 66435 IC50 > 300000 nM T16347 D03TTQ 6296 IC50 = 3900 nM T16347 D07HBX 338 Ki = 19400000 nM T16347 D0K8KX 5280343 IC50 = 23300 nM T16347 D0P2CS 9409 IC50 = 1300 nM T16347 D0W8WB 2353 IC50 = 67000 nM T16347 D0Z2RA 5944 IC50 = 3600 nM T16347 D04SLF 9903 IC50 = 12740 nM T16347 D0O3QW 9917968 IC50 = 1000 nM T16347 D0QR5G 2355 IC50 = 2.53 ug.mL-1 T16347 D0T8QB 14982 IC50 > 100000 nM T16347 D0U3EP 445154 IC50 > 1000000 nM T16347 D0I2AN 86298439 IC50 = 2290 nM T16347 D06WBE 157049 IC50 = 384 nM T16347 D0DN1I 23080446 Ki = 220 nM T16347 CSI0D4 355 IC50 = 250000 nM T16347 CV5K8P 1521 Ki = 8300 nM T16347 C6COK9 1854 Ki = 22000 nM T16347 C7AGI4 2741 IC50 > 1000000 nM T16347 CEXU05 3383 IC50 = 600000 nM T16347 CQ0D8J 3469 IC50 > 100000 nM T16347 C4VM6O 4964 Ki = 43000 nM T16347 CQX7W5 4965 Ki = 128000 nM T16347 CG0FD6 4966 Ki = 193000 nM T16347 CU7AC1 6259 Ki = 81000 nM T16347 CYZ1D6 6585 Ki = 17000000 nM T16347 C3RJ7D 6844 IC50 = 850000 nM T16347 C74YCT 7103 IC50 = 162181009.7 nM T16347 C2JK3W 7104 IC50 > 1000000 nM T16347 CHG8L5 7322 IC50 > 1000000 nM T16347 CJKY76 7420 IC50 > 100000 nM T16347 CEVL63 9348 IC50 = 859000 nM T16347 CJBC76 10710 IC50 = 1500000 nM T16347 CU94VJ 11393 IC50 = 3500000 nM T16347 CU5WV4 11914 IC50 = 5500000 nM T16347 C28BQV 11915 IC50 = 2700000 nM T16347 C52KJE 14749 IC50 = 26000 nM T16347 CZ5O2D 15587 IC50 = 210000 nM T16347 C05CMQ 20353 IC50 = 25050 nM T16347 CQ7GE6 20834 IC50 = 1580 nM T16347 CE3U1F 26218 IC50 = 8050 nM T16347 CS73YX 33258 IC50 = 33000 nM T16347 CKD90R 38384 Ki = 173000 nM T16347 CO19PJ 55294 Ki = 6200 nM T16347 CW68ZS 61672 IC50 = 46 nM T16347 C74KLR 65235 IC50 = 150000 nM T16347 CUAV28 66834 Ki = 1400000 nM T16347 CK2VX3 66840 Ki = 195000 nM T16347 CA74FI 66900 IC50 = 910000 nM T16347 CV1X5G 67282 Ki = 14000 nM T16347 CDZI90 67584 IC50 = 1279000 nM T16347 CK4HU2 67658 IC50 > 1000000 nM T16347 C2H0JD 68066 IC50 = 63500 nM T16347 C7LCW5 69179 Ki = 25000 nM T16347 CO0JW2 69226 IC50 > 1000000 nM T16347 CD6SZ4 69748 IC50 > 500000 nM T16347 CYI58D 72185 IC50 = 12000 nM T16347 C7UMO3 72908 IC50 = 24590 nM T16347 CU75FJ 73062 IC50 = 20200 nM T16347 CKB4R0 73145 IC50 > 100000 nM T16347 CXJV17 73157 IC50 = 800 nM T16347 CKH0W1 73170 IC50 = 19260 nM T16347 C7R2OM 73412 IC50 = 12380 nM T16347 CFM6N8 73846 Ki = 79000 nM T16347 C2SCG6 73863 IC50 = 390000 nM T16347 CAX8Y2 74248 IC50 = 28000000 nM T16347 CIQO73 74974 Ki = 31000 nM T16347 C3Y6ZR 76658 IC50 > 200000 nM T16347 C7X0LB 77694 IC50 = 950000 nM T16347 C4D3ZC 79628 IC50 > 1000000 nM T16347 C7GTI4 81312 Ki = 3000000 nM T16347 CV5C3X 85405 IC50 = 354200 nM T16347 C5Z6KQ 86860 IC50 = 27000 nM T16347 CQ1RK5 87112 IC50 = 73000 nM T16347 CBVH30 92794 IC50 = 17500 nM T16347 C31IYR 92900 IC50 = 4440 nM T16347 C7LH1Z 95168 IC50 = 23600 nM T16347 C4S0UL 96582 IC50 > 10000 nM T16347 C14SVF 96749 Ki = 56000 nM T16347 CHF2E5 101761 IC50 = 9600 nM T16347 CUNH62 112056 IC50 = 5700000 nM T16347 C1TNJ0 120248 Ki = 380000 nM T16347 CD1JI7 124052 IC50 = 73400 nM T16347 C57VPM 129362 IC50 > 60000 nM T16347 CYF95X 129597 IC50 = 10000 nM T16347 CB0L4N 136414 IC50 = 61659500.19 nM T16347 C1MSI6 145761 IC50 = 1700000 nM T16347 C2FIH6 149160 IC50 > 10000 nM T16347 CRC4A0 149161 IC50 > 10000 nM T16347 CV9PX7 150081 IC50 > 10000 nM T16347 C1JF4U 151202 IC50 = 21500 nM T16347 C8VIR1 151940 IC50 = 2700000 nM T16347 CJ8E3C 159087 IC50 = 130000 nM T16347 C5X1YU 160254 IC50 = 33500 nM T16347 CV8A4D 163098 IC50 > 30000 nM T16347 CW8K1N 168928 IC50 > 20000 nM T16347 C0CX1A 189061 IC50 = 45600 nM T16347 CKEU36 194183 IC50 > 30000 nM T16347 CND73T 195173 IC50 = 39200 nM T16347 C83JYG 195652 IC50 = 24200 nM T16347 CH1FS8 197678 IC50 = 5000 nM T16347 CGPH69 221862 IC50 = 60255958.61 nM T16347 CLO9Q8 231868 IC50 = 11990 nM T16347 C6KSA8 242834 IC50 = 707945784.4 nM T16347 C8OHY9 254021 IC50 > 30000 nM T16347 C10MJX 259218 Ki = 10330 nM T16347 CCEG90 259329 IC50 = 62400 nM T16347 CVLC68 268455 IC50 = 149000 nM T16347 CPL6E4 272516 IC50 = 34880 nM T16347 CL15BT 321979 Ki = 14000 nM T16347 CFL2Q5 339496 IC50 = 1160000 nM T16347 CI3K5N 378911 IC50 > 10000 nM T16347 C7BAY8 379075 IC50 > 10000 nM T16347 C5Q7BU 386231 IC50 > 100000 nM T16347 C02WIT 388306 IC50 > 10000 nM T16347 C7HME8 439246 IC50 = 130100 nM T16347 C0DT9W 439616 IC50 = 4900000 nM T16347 C29OPT 441958 IC50 = 74100 nM T16347 C6WI0Q 442431 IC50 = 56500 nM T16347 CWV1I2 442774 IC50 = 5000 nM T16347 C1PJ5Z 443023 IC50 = 15010 nM T16347 CF7Q0W 443028 IC50 = 16820 nM T16347 CONR62 444765 Ki = 14000 nM T16347 C9B3YM 444766 Ki = 230 nM T16347 CQN15I 445785 Ki = 220 nM T16347 CH01QN 446464 Ki = 2000 nM T16347 CU6R9H 446662 IC50 = 26000 nM T16347 CM0IQ3 446665 Ki = 1500 nM T16347 C5Y3DJ 446871 Ki = 1100 nM T16347 CX1LO8 447392 Ki = 1096.48 nM T16347 CE5B6L 447410 Ki = 19.95 nM T16347 CF18DI 447411 Ki = 24000 nM T16347 C5MF7I 447695 Ki = 17000 nM T16347 CO7IJ1 447968 Ki = 3200 nM T16347 C4I1LX 447994 Ki = 6309.57 nM T16347 CJ4M3B 448021 IC50 = 16 nM T16347 CW5YV0 448024 IC50 = 12 nM T16347 C6STF5 448214 Ki = 9000 nM T16347 CL03SZ 448662 IC50 = 2000 nM T16347 CWK8E7 449162 IC50 = 920 nM T16347 CX6S0R 455821 IC50 = 10.42 ug.mL-1 T16347 C15JUM 463777 IC50 = 28000 nM T16347 C7GU8T 470607 IC50 = 2330 nM T16347 CV0ZD5 480783 IC50 = 9300 nM T16347 CV03EX 480802 IC50 = 550 nM T16347 CHQ39C 483758 IC50 = 40000 nM T16347 CF9T4V 484588 IC50 = 62400 nM T16347 CDI64A 489941 Ki = 8000 nM T16347 CY8HW5 489944 Ki = 7100 nM T16347 CEM6N5 493415 IC50 = 20000 nM T16347 C84QRW 493418 IC50 = 20000 nM T16347 CA5JR0 503731 IC50 = 71200 nM T16347 CGH3A2 510684 IC50 = 20000 nM T16347 CS3PI2 516996 IC50 = 5290 nM T16347 C5T4LR 520927 IC50 > 1000000 nM T16347 CKG5C2 522129 IC50 = 25000 nM T16347 CBT0U1 584714 IC50 = 150000 nM T16347 CK9B6W 585053 Ki = 1000000 nM T16347 C2NM3I 588083 Ki = 17500000 nM T16347 C1C3ZG 591773 IC50 > 200000 nM T16347 CCA8H2 594762 IC50 = 29110 nM T16347 CHX62Y 598522 IC50 > 30000 nM T16347 CG2LA4 606638 IC50 = 18000 nM T16347 CMZ3H1 614309 IC50 = 20000 nM T16347 CFN60B 637141 IC50 = 11500 nM T16347 CO2Z1S 637195 IC50 = 50020 nM T16347 CZ0AH3 638278 IC50 > 60000 nM T16347 C9L2WJ 641672 IC50 > 30000 nM T16347 CJ6QK3 643007 IC50 = 1.97 ug.mL-1 T16347 CTB7Y4 648231 IC50 = 65000 nM T16347 CGVB58 668081 IC50 = 11.55 ug.mL-1 T16347 C9FA1S 688710 IC50 = 20000 nM T16347 CJY09B 688711 IC50 = 22000 nM T16347 CSH95Z 688893 IC50 = 55000 nM T16347 C5GHU8 735928 IC50 > 1000000 nM T16347 CX18QE 767146 Ki = 3000 nM T16347 CXYV26 849731 IC50 > 10000 nM T16347 CU1A3R 884226 Ki = 7100 nM T16347 C4COH2 890791 IC50 = 14000 nM T16347 CELG48 998012 IC50 = 19270 nM T16347 CJ3K7L 1006953 IC50 = 25000 nM T16347 CN48LB 1015488 IC50 = 35000 nM T16347 CA8OH9 1019926 IC50 = 18540 nM T16347 CE4HM8 1032885 IC50 = 38800 nM T16347 C2OS9P 1098316 IC50 = 14000 nM T16347 CPN82R 1101867 IC50 = 15000 nM T16347 CJ90PO 1159989 IC50 = 38000 nM T16347 CCXP42 1201110 IC50 = 171000 nM T16347 CXNA13 1201165 IC50 = 86800 nM T16347 C0B3ZE 1201317 IC50 = 54100 nM T16347 CH82ZT 1201321 IC50 = 43100 nM T16347 CP7AH1 1208911 IC50 = 11000 nM T16347 CS1L6Q 1230239 IC50 = 4400 nM T16347 CKWD10 1249523 IC50 = 42000 nM T16347 C1D5NJ 1252884 IC50 = 23000 nM T16347 CW6VR9 1268078 IC50 = 91000 nM T16347 CE4YD2 1271283 IC50 = 34400 nM T16347 C1RHZ7 1330090 IC50 = 43000 nM T16347 C70SGI 1334376 IC50 = 1700 nM T16347 CXY1W8 1363495 IC50 = 11000 nM T16347 CMQ95J 1363496 IC50 = 11000 nM T16347 CBN5Y6 1367261 Ki = 20400 nM T16347 CV1QW2 1379873 IC50 = 18970 nM T16347 C6UZ1A 1383990 IC50 = 56000 nM T16347 CK94XG 1403665 IC50 = 14000 nM T16347 CPF4S9 1480751 IC50 = 25000 nM T16347 CGEW23 1526715 IC50 = 14680 nM T16347 C9Q4MJ 1526752 IC50 = 2270 nM T16347 C71RFL 1558734 IC50 = 22000 nM T16347 CD9OU5 1613011 IC50 = 35000 nM T16347 CCW1J7 1778937 IC50 = 21600 nM T16347 C6ZW8Y 1789777 IC50 = 12520 nM T16347 CCQ3S1 1854415 IC50 = 12000 nM T16347 CRC9X4 1902393 IC50 = 3200 nM T16347 CI0H6E 1908130 IC50 = 27000 nM T16347 CU0A3X 1921859 IC50 > 100000 nM T16347 C4RH2W 1933357 IC50 > 100000 nM T16347 C7LNT5 1967843 IC50 = 2600 nM T16347 C7CTM1 1979301 IC50 = 1850 nM T16347 CR51YM 2015276 IC50 = 6580 nM T16347 C57QFS 2063329 IC50 = 48977881.94 nM T16347 C3ZLD4 2261820 Ki = 1800 nM T16347 CQZ47H 2710079 IC50 = 69000 nM T16347 C3X1KJ 2711328 IC50 = 74000 nM T16347 CF5BV8 2734086 IC50 = 3850 nM T16347 CFK5Z0 2765033 IC50 > 100000 nM T16347 CQOC30 2765069 IC50 > 120000 nM T16347 CIV1E3 2775086 IC50 > 500000 nM T16347 CPG92K 2819267 IC50 = 63900 nM T16347 CB7OS1 2964738 IC50 = 120000 nM T16347 CYRQ35 2987937 IC50 = 8500 nM T16347 CI1X7Q 3014027 IC50 > 4000000 nM T16347 C4X2BE 3163277 IC50 = 8200 nM T16347 CLX1P8 3241797 IC50 = 77000 nM T16347 C3NL9W 3246406 IC50 = 96700 nM T16347 C0KA3Q 3433760 IC50 > 100000 nM T16347 C4LDC9 3830513 Ki = 92000 nM T16347 C3XM5J 3955344 IC50 = 40000 nM T16347 CA35NM 4171145 IC50 = 30000 nM T16347 CHYD58 4369034 IC50 < 1 nM T16347 C6O9LC 4369451 IC50 = 2470 nM T16347 CFH48I 4469997 Ki = 22 nM T16347 CJZ02Q 4470789 Ki = 76 nM T16347 C12CHL 4470793 Ki = 630.96 nM T16347 CO3PG6 4471649 IC50 = 87000 nM T16347 C8SZY6 4584157 IC50 > 100000 nM T16347 C0SZ5T 4626075 IC50 = 4100 nM T16347 C35LZP 4774445 Ki = 1000 nM T16347 C64EDY 4779151 IC50 = 72443596.01 nM T16347 CP6F3M 5011693 IC50 = 48000 nM T16347 CI9X0D 5214210 IC50 = 1510000 nM T16347 CBWK73 5280435 IC50 = 32600 nM T16347 C81FUM 5280633 IC50 = 31600 nM T16347 CU0E5R 5281219 IC50 = 20600 nM T16347 CG0C4J 5281255 IC50 = 27300 nM T16347 C3ZJ8U 5281609 IC50 = 9600 nM T16347 CZQ27P 5281631 IC50 = 149900 nM T16347 C0D3PO 5281671 IC50 = 10320 nM T16347 CGS9B0 5281780 IC50 = 41500 nM T16347 C2F8GX 5287526 Ki = 169.82 nM T16347 CUWZ35 5288267 Ki = 2.4 nM T16347 C0YCX9 5315126 IC50 = 21500 nM T16347 C4CKU6 5315396 IC50 = 26700 nM T16347 CRD56H 5316802 IC50 = 450 nM T16347 CTJ29I 5317563 Ki = 19900 nM T16347 CUQ0S8 5317652 IC50 = 66300 nM T16347 C0UKZ1 5317756 IC50 = 183900 nM T16347 CBX74L 5317764 IC50 = 58700 nM T16347 CP1F2V 5318990 IC50 = 59500 nM T16347 C94XGK 5318993 IC50 = 6000 nM T16347 C7J6ZH 5319000 IC50 = 54500 nM T16347 CC85JG 5324104 Ki = 7070 nM T16347 CQK4M1 5327152 IC50 = 42500 nM T16347 CPM09B 5327156 IC50 = 4800 nM T16347 CA39QI 5327157 IC50 = 33500 nM T16347 CP08UL 5327158 IC50 = 2500 nM T16347 CPN83Z 5358846 IC50 = 3600 nM T16347 C6ZO0N 5372312 IC50 = 5700 nM T16347 CH64SX 5382771 IC50 = 23000 nM T16347 CAZ19U 5383850 IC50 = 107000 nM T16347 CZGP09 5441538 IC50 = 19300 nM T16347 CH5OM1 5463917 IC50 = 30800 nM T16347 CSN0W5 5481949 IC50 = 1480 nM T16347 CWS5X0 5481970 IC50 = 5180 nM T16347 C98YJF 5487298 IC50 = 27900 nM T16347 CS2KQ6 5490139 IC50 = 41500 nM T16347 C3EPL0 5605148 IC50 = 68000 nM T16347 CI4U9Z 5711223 IC50 > 60000 nM T16347 C0PCZ3 5932584 IC50 = 420 nM T16347 C95HVU 5939774 IC50 = 64000 nM T16347 CU65JT 5998084 IC50 = 1800 nM T16347 CD1Z2I 6058371 IC50 = 14220 nM T16347 CY81DG 6118992 Ki = 170 nM T16347 C14LAC 6161281 IC50 = 460 nM T16347 CR6O8V 6166563 IC50 = 2200 nM T16347 C54BYS 6172647 IC50 = 34000 nM T16347 CWT69J 6178946 IC50 = 3090000 nM T16347 CYI5R1 6274486 IC50 = 590 nM T16347 CAE1T0 6377130 IC50 = 170000 nM T16347 CZ75UC 6438503 IC50 = 2.47 ug.mL-1 T16347 C1HZJ2 6438825 IC50 = 21500 nM T16347 C3EI9B 6441564 IC50 = 9900 nM T16347 CD51MJ 6442675 IC50 > 50000 nM T16347 C0KUG9 6442843 IC50 = 1.49 nM T16347 C45QJF 6474309 IC50 = 59400 nM T16347 CSA24L 6474310 IC50 = 37900 nM T16347 CR7ZY0 6474640 IC50 = 35400 nM T16347 C5WM0L 6478429 IC50 > 24000 nM T16347 CUO1S6 6479088 IC50 = 1.67 ug.mL-1 T16347 C9OV3N 6504357 IC50 = 63800 nM T16347 C2ML1B 6521442 IC50 = 26600 nM T16347 CXL68K 6548074 IC50 = 26300 nM T16347 CF48XG 6914659 IC50 = 6100 nM T16347 CZU0N8 7158830 IC50 > 100000 nM T16347 CV0FA1 7330517 IC50 = 29200 nM T16347 CQ0H9V 7729033 IC50 = 158490 nM T16347 CM07FD 7946130 IC50 = 263000 nM T16347 CLH37Y 7947894 IC50 = 144540 nM T16347 COBT25 8002021 IC50 = 1258930 nM T16347 C9QPV8 9448597 IC50 = 123030 nM T16347 CBH2X6 9547919 IC50 = 1750 nM T16347 CSO84R 9547958 Ki = 300 nM T16347 CPE73S 9547959 Ki = 1300 nM T16347 CHC9A2 9547975 Ki = 160000 nM T16347 CUS63A 9549198 Ki = 1.7 nM T16347 C3RK8Y 9549199 IC50 = 270 nM T16347 C82XTA 9797177 Ki = 12000 nM T16347 CHI48L 9798666 IC50 = 43900 nM T16347 CEM40C 9807672 IC50 = 74 nM T16347 C4H0IZ 9807792 IC50 = 80 nM T16347 CCL4Y9 9808144 IC50 = 1200 nM T16347 C1R2KI 9808280 IC50 = 27542287.03 nM T16347 CG6W0B 9809625 Ki = 8400 nM T16347 C0GN6A 9809675 IC50 = 53 nM T16347 CW5P3S 9810271 IC50 = 25 nM T16347 CVYN58 9810403 IC50 = 61 nM T16347 CGK46C 9810983 IC50 = 4600 nM T16347 CV94PD 9817302 Ki = 14000 nM T16347 CCJY82 9819655 Ki = 12882.5 nM T16347 C18MYG 9820314 Ki = 1000 nM T16347 C9TMX5 9821764 Ki = 700 nM T16347 C3K4RH 9823082 IC50 = 1150 nM T16347 CX2C9V 9825492 Ki = 18 nM T16347 CB2IT7 9826909 IC50 = 700 nM T16347 C6ILQ0 9829174 IC50 = 370 nM T16347 C9T8XN 9829273 IC50 = 106 nM T16347 C9KEW5 9830016 IC50 = 28 nM T16347 C4VZQ8 9830376 IC50 = 77 nM T16347 CIY94Z 9830685 IC50 = 42.66 nM T16347 CR5U9X 9830938 IC50 = 53.7 nM T16347 CBGP53 9830970 IC50 = 52 nM T16347 CWN24D 9831951 IC50 = 30 nM T16347 CJ5CS1 9834233 IC50 = 190000 nM T16347 C2DJ1Y 9836432 Ki = 93000 nM T16347 C2O1IN 9838736 Ki = 1000 nM T16347 CBFZ26 9839539 Ki = 4466.84 nM T16347 CW0G3C 9839618 Ki = 7943.28 nM T16347 C79LEI 9840805 IC50 = 30900 nM T16347 CH2QD7 9842328 IC50 = 3981071.71 nM T16347 C05FGO 9842446 IC50 = 230 nM T16347 CJCO34 9843618 Ki = 5700 nM T16347 COL5Q6 9847403 IC50 = 1400 nM T16347 CQT1A6 9848618 IC50 = 120 nM T16347 C1DMN7 9850223 IC50 = 29800 nM T16347 CUN43C 9850346 IC50 = 1600 nM T16347 CK28BN 9850783 IC50 = 75 nM T16347 C6C8YD 9851148 IC50 = 39 nM T16347 CRP5J3 9852025 IC50 = 58 nM T16347 CI7MW0 9852185 Ki = 190 nM T16347 C49AFB 9861219 IC50 = 23500 nM T16347 CKDB51 9863049 IC50 = 1100 nM T16347 C4PQJ7 9863691 Ki = 1000 nM T16347 C54CTK 9863756 IC50 = 18200 nM T16347 C86MNV 9864366 Ki = 270 nM T16347 C5YIN8 9865448 IC50 = 12589254.12 nM T16347 C06VSQ 9867075 IC50 = 480 nM T16347 C1ECT8 9867205 IC50 = 8000 nM T16347 C1IR5A 9867355 IC50 = 540 nM T16347 C0NG3L 9871566 Ki = 1500 nM T16347 CWIJ57 9873352 IC50 = 38 nM T16347 C4HV0Y 9873483 IC50 = 85.11 nM T16347 C30SGW 9873553 IC50 = 56 nM T16347 CR6D0J 9873582 IC50 = 34 nM T16347 C4BE0F 9874843 IC50 = 83 nM T16347 C5SQ2K 9876301 IC50 = 4800 nM T16347 CJIZ31 9878547 IC50 = 25600 nM T16347 C34BQA 9882296 Ki = 1995.26 nM T16347 CWP06Z 9882419 IC50 > 30000 nM T16347 CXO9K1 9884811 Ki = 25000 nM T16347 C46QVW 9886299 Ki = 25703.96 nM T16347 CDG61K 9894866 IC50 = 190546071.8 nM T16347 CUL4E2 9895320 IC50 = 29 nM T16347 C3A5DF 9895569 IC50 = 28 nM T16347 CI59PS 9895735 IC50 = 28 nM T16347 C8SB2Q 9895791 IC50 = 52 nM T16347 C9XA0I 9895792 IC50 = 190 nM T16347 CS3M5T 9896246 IC50 = 38 nM T16347 CPR9S3 9896840 IC50 = 74 nM T16347 C5DYS8 9897771 IC50 = 13800 nM T16347 C2JCM5 9902742 IC50 = 18000 nM T16347 C5Z8VD 9905439 Ki = 2187.76 nM T16347 CDB50K 9905786 Ki = 4677.35 nM T16347 C1XP7G 9908778 Ki = 15848.93 nM T16347 CY2UE8 9909415 IC50 = 330 nM T16347 C5BYE4 9914773 IC50 = 270 nM T16347 C63YNT 9914774 IC50 = 320 nM T16347 C53MUC 9915344 IC50 = 1300 nM T16347 C1Q3WM 9915604 IC50 = 650 nM T16347 C6JZH3 9916414 IC50 = 148300 nM T16347 C8N2JF 9917026 IC50 = 100 nM T16347 CD0S9U 9917827 IC50 = 24 nM T16347 C6YF5L 9918081 Ki = 39.81 nM T16347 CRL95K 9923781 Ki = 39000 nM T16347 CU7G8V 9926545 Ki = 6025.6 nM T16347 CXD2Y6 9926586 IC50 > 30000 nM T16347 COX2J8 9930943 IC50 = 5000 nM T16347 CD1ZT3 9931427 Ki = 1800 nM T16347 CC29PS 9933616 IC50 = 800 nM T16347 CP5GK3 9949406 IC50 = 1300 nM T16347 C7EA3R 9955674 IC50 = 380 nM T16347 C02YNS 9956737 IC50 = 2000 nM T16347 CJCB98 9958642 IC50 = 1400 nM T16347 CTJZ08 9959737 IC50 = 77 nM T16347 C2YS6H 9960407 IC50 = 320 nM T16347 C21HPD 9960929 IC50 = 28.84 nM T16347 CWFI76 9961320 IC50 = 25 nM T16347 C93ANO 9961383 IC50 = 284 nM T16347 C1BE5J 9970370 IC50 = 8200 nM T16347 CA75NG 9985013 IC50 = 1700 nM T16347 CQYC90 9998434 Ki = 79432.82 nM T16347 C86RXM 10001604 IC50 = 90500 nM T16347 CCG8T2 10009628 IC50 = 600 nM T16347 CO7T0B 10009840 IC50 = 40 nM T16347 CQA9G0 10010762 IC50 = 3200 nM T16347 COIB51 10018011 IC50 = 115000 nM T16347 C6GN0L 10022050 IC50 = 1.43 ug.mL-1 T16347 CGO91A 10029121 IC50 < 10000 nM T16347 CEJ6L0 10048747 IC50 = 4300 nM T16347 CKS9R4 10049789 IC50 > 24000 nM T16347 C4GNQ6 10055128 Ki = 3200 nM T16347 C6C9DL 10055263 Ki = 63.1 nM T16347 C1BVS2 10055383 Ki = 590 nM T16347 CD1MX4 10055524 IC50 = 131825673.9 nM T16347 C2E5OK 10072839 IC50 > 24000 nM T16347 CHGX49 10075681 IC50 = 42700 nM T16347 CT64NM 10077494 IC50 = 13000 nM T16347 CL78RJ 10078618 IC50 = 350 nM T16347 C4JT9D 10087747 IC50 = 4300 nM T16347 CK35NL 10090732 IC50 = 39600 nM T16347 CF83UC 10094446 IC50 = 53000 nM T16347 CTNK21 10101005 Ki = 1800 nM T16347 CV5M7L 10101397 IC50 = 21700 nM T16347 CJF2W6 10108804 IC50 = 5200 nM T16347 C3Y8QT 10119338 IC50 = 2000 nM T16347 C53KYA 10145907 Ki = 316.23 nM T16347 CPES42 10146934 IC50 = 5 nM T16347 CKB1Q8 10150793 IC50 = 4500 nM T16347 CM2CK3 10167662 IC50 = 39 nM T16347 CSO2C9 10168739 IC50 = 3 nM T16347 C0URF3 10169038 IC50 = 11 nM T16347 CYV93G 10172292 IC50 = 6200 nM T16347 CRUV90 10184204 IC50 = 2250 nM T16347 CUV6M1 10198815 IC50 = 12000 nM T16347 CZ7A6O 10206788 IC50 = 1950 nM T16347 C95BCN 10211112 Ki = 630.96 nM T16347 CJEW67 10211810 IC50 = 18 nM T16347 CZ8JC5 10212468 IC50 = 220 nM T16347 CJT84V 10220129 Ki = 1100000 nM T16347 C7U0ZQ 10226739 IC50 = 4400 nM T16347 C95ILX 10237678 IC50 = 33000 nM T16347 CHV18Y 10248262 IC50 > 30000 nM T16347 CBD3E1 10250245 Ki = 50118.72 nM T16347 CWQB59 10251757 Ki = 11000 nM T16347 CFQZ83 10252345 IC50 = 3890 nM T16347 CEJN86 10253374 IC50 = 24000 nM T16347 CSX9F6 10253609 IC50 > 24000 nM T16347 C3A8JL 10256983 IC50 = 4200 nM T16347 CH45KB 10258785 Ki = 2.4 nM T16347 C0RD1X 10260174 Ki = 26 nM T16347 C9R7HY 10263317 IC50 = 19000 nM T16347 CXA6K2 10298514 IC50 = 2200 nM T16347 CVP6R4 10300190 IC50 = 1180 nM T16347 C0O6CP 10305270 IC50 = 69 nM T16347 CC30ZA 10305301 Ki = 120 nM T16347 CPGO28 10325639 IC50 > 24000 nM T16347 CZ90BA 10325640 IC50 > 19000 nM T16347 C38ZVN 10327524 IC50 = 58200 nM T16347 C9N6OP 10328286 IC50 = 4400 nM T16347 CX1YP3 10332717 IC50 = 112000 nM T16347 C7IN9O 10340643 IC50 = 10000000 nM T16347 C9I7WV 10348668 IC50 = 4580 nM T16347 C73RHZ 10348783 IC50 = 470 nM T16347 CP6JD4 10357078 Ki = 47000 nM T16347 C8A6EM 10364207 Ki = 2100 nM T16347 C0D9QX 10372989 Ki = 160 nM T16347 CR9FX4 10392218 IC50 = 56000 nM T16347 C4M3AW 10397889 IC50 = 10130 nM T16347 CRW54P 10408069 IC50 = 72900 nM T16347 CA6ZE1 10408212 IC50 > 30000 nM T16347 CH70EY 10414856 IC50 = 4500 nM T16347 CQ79JD 10420098 IC50 > 50000 nM T16347 C5T0GC 10422621 IC50 = 35000 nM T16347 CY2TU6 10426622 IC50 = 53000 nM T16347 C41YFU 10429577 Ki = 79432.82 nM T16347 C4J8LM 10433041 IC50 = 19000 nM T16347 CV4ZJ6 10434105 IC50 = 1480 nM T16347 CI3VG8 10439203 Ki = 670 nM T16347 C3KEQ2 10439508 IC50 = 23 nM T16347 CA7N0T 10439869 Ki = 15200 nM T16347 C05SVE 10444314 IC50 = 320 nM T16347 CP70SY 10453228 Ki = 6309.57 nM T16347 C4HE0C 10458201 IC50 = 29000 nM T16347 C6A5PJ 10468556 Ki = 93000 nM T16347 C9MXL0 10474985 Ki = 15848.93 nM T16347 CGA27K 10479064 IC50 = 63095734.45 nM T16347 CZ50LG 10485602 IC50 = 5 nM T16347 C73DGE 10485872 IC50 = 1000 nM T16347 C2TYE0 10499446 IC50 = 18000 nM T16347 CX37AL 10500598 IC50 = 740 nM T16347 CH14JZ 10504580 IC50 = 13000 nM T16347 C7IN2X 10506471 IC50 = 478630092.3 nM T16347 CCJV57 10506617 IC50 = 109.65 nM T16347 C9G6BW 10506650 IC50 = 1550 nM T16347 CEC76W 10507016 IC50 = 169.82 nM T16347 C6MBX9 10507672 IC50 = 54.95 nM T16347 CY93MH 10513846 IC50 = 860 nM T16347 CK5F4M 10517813 IC50 > 30000 nM T16347 CZA2C3 10521037 IC50 = 9000 nM T16347 CS1VH8 10529709 IC50 = 360 nM T16347 C0FE7M 10530210 IC50 = 2860 nM T16347 C8A7EO 10531082 IC50 = 229.09 nM T16347 C6C8HK 10531763 IC50 = 340 nM T16347 C7LKX3 10542808 IC50 = 62700 nM T16347 C1H7OE 10546338 IC50 = 700 nM T16347 CD70YL 10547545 IC50 = 912.01 nM T16347 C0OT9Z 10548559 IC50 = 93325430.08 nM T16347 CYZ4M0 10548992 IC50 = 2190 nM T16347 CC91GX 10551711 IC50 = 275422870.3 nM T16347 C6TOK7 10553086 IC50 = 970 nM T16347 C8YN1K 10553616 IC50 = 169.82 nM T16347 CLFA64 10553635 IC50 = 48000 nM T16347 C9L7NF 10554119 IC50 = 100 nM T16347 C8VSC2 10554409 IC50 = 290 nM T16347 C7JQS4 10554508 IC50 = 602559586.1 nM T16347 C58EUG 10555074 IC50 = 32 nM T16347 COUA78 10555076 IC50 = 52 nM T16347 C7SL4Z 10574839 IC50 = 288403150.3 nM T16347 CX6PD4 10578752 IC50 = 120.23 nM T16347 C0DQ8N 10582552 IC50 = 18000 nM T16347 CM45AC 10599143 IC50 = 510 nM T16347 CT8JC1 10601104 IC50 = 457.09 nM T16347 CBW5G6 10602493 IC50 = 220 nM T16347 CG7W0T 10622249 IC50 = 575.44 nM T16347 C9S1PA 10626001 IC50 = 1160 nM T16347 CMYB73 10626244 IC50 = 158.49 nM T16347 CS3GW0 10626561 IC50 = 82 nM T16347 C2IBJ7 10627951 IC50 = 520 nM T16347 C3QNE6 10629121 IC50 = 11 nM T16347 CVOU27 10636947 IC50 = 19952623.15 nM T16347 C5GK3L 10638003 IC50 = 1000 nM T16347 C8D7SU 10642019 IC50 = 165958690.7 nM T16347 COTK63 10643491 IC50 = 10500 nM T16347 C0LOG3 10645149 IC50 = 1071.52 nM T16347 CIU60C 10648773 IC50 = 440 nM T16347 CMG58E 10649372 IC50 = 398.11 nM T16347 C37UKN 10649445 IC50 = 407380277.8 nM T16347 CX8CK6 10650640 IC50 = 831763771.1 nM T16347 C1OQ2N 10651932 IC50 = 40 nM T16347 CHDL03 10673144 IC50 = 1100 nM T16347 C6PO0E 10673660 IC50 = 590 nM T16347 C8DW6I 10674946 IC50 = 370 nM T16347 C3NJY2 10675095 IC50 = 120 nM T16347 CZTN01 10675368 IC50 = 390 nM T16347 CL59UR 10675666 IC50 = 120 nM T16347 CM51YT 10675911 IC50 = 46.77 nM T16347 C5QZ0U 10676857 IC50 = 54 nM T16347 C6YNV0 10685375 IC50 = 7300 nM T16347 CKQ7B9 10697392 IC50 = 436515832.2 nM T16347 CNX4Z6 10697668 IC50 = 680 nM T16347 CW1OK8 10698324 IC50 = 120 nM T16347 C0K2CU 10706701 IC50 = 175000 nM T16347 CI93LN 10719718 IC50 = 354 nM T16347 CZ9TW3 10719937 IC50 = 109.65 nM T16347 C1YO7J 10721150 IC50 = 588843655.4 nM T16347 C7JS3X 10721373 IC50 = 446.68 nM T16347 CC3RI0 10721544 IC50 = 5970 nM T16347 CP4MW9 10734041 IC50 = 31622776.6 nM T16347 CH85LK 10744488 IC50 = 510 nM T16347 C5OML1 10744622 IC50 = 350 nM T16347 C7ZT2I 10745063 IC50 = 130 nM T16347 CGO80Z 10745191 IC50 = 1160 nM T16347 C0UT5L 10745907 IC50 = 70.79 nM T16347 CWK87I 10746742 IC50 = 160 nM T16347 C05PEI 10746943 IC50 = 25 nM T16347 C8YR9K 10747376 IC50 = 290 nM T16347 C31IOZ 10757624 IC50 = 16000 nM T16347 CW7LG8 10765880 IC50 = 1320 nM T16347 CJOC32 10767413 IC50 = 912.01 nM T16347 CE8N5Y 10767785 IC50 = 170 nM T16347 C9YQ4C 10768812 IC50 = 95.5 nM T16347 C4ZGB8 10770595 IC50 = 145 nM T16347 CCI4U6 10777789 IC50 = 3300 nM T16347 CR4Z7G 10783655 IC50 = 3162277.66 nM T16347 CK9J4E 10783699 IC50 > 30000 nM T16347 CHK60Z 10790583 IC50 = 1071.52 nM T16347 C92DNK 10791327 IC50 = 1300 nM T16347 CYH14L 10792205 IC50 = 213796209 nM T16347 CO97SN 10794070 Ki = 1210 nM T16347 C1CNY2 10805901 IC50 = 19000 nM T16347 C8RY6F 10814471 IC50 = 900 nM T16347 CP2OG3 10817657 IC50 = 128.82 nM T16347 C5WCV7 10819036 IC50 = 44 nM T16347 C64EDJ 10819125 IC50 = 180 nM T16347 C4GZK3 10839919 IC50 = 360 nM T16347 CGO41K 10840654 IC50 = 384 nM T16347 C8MBX4 10840751 IC50 = 140 nM T16347 C1LN7F 10841392 IC50 = 100 nM T16347 C30VWD 10859452 Ki = 10964.78 nM T16347 C1T3PD 10864326 Ki = 1200 nM T16347 C7HF1Z 10875237 Ki = 15848.93 nM T16347 C13WSN 10881804 IC50 = 44300 nM T16347 COV48X 10882941 Ki = 1100 nM T16347 CC65TP 10890191 IC50 = 20000000 nM T16347 C2AVQ5 10892825 Ki = 12589.25 nM T16347 C0N4FE 10903324 Ki = 8912.51 nM T16347 C4GA1U 10912909 Ki = 12940 nM T16347 C92AER 10914619 IC50 > 30000 nM T16347 CZ53SY 10917594 Ki = 5900 nM T16347 CWB8C1 10919218 Ki = 2000 nM T16347 CZTX36 10928920 Ki = 16000 nM T16347 C87NWE 10930296 Ki = 1600 nM T16347 CY0I6J 10935182 Ki = 12882.5 nM T16347 CA2EU5 10945946 Ki = 12000 nM T16347 C4IY6P 10956980 Ki = 1288.25 nM T16347 CLSK91 10959075 Ki = 7943.28 nM T16347 CLK0Q5 10967229 IC50 = 2800000 nM T16347 C3YWN8 10975947 IC50 > 80000 nM T16347 CB6Z1K 10981284 Ki = 900 nM T16347 C3BG6Y 10981976 Ki = 7300 nM T16347 C7G1IP 10988114 IC50 = 12000000 nM T16347 CTB71O 10998288 Ki = 158489.32 nM T16347 CLT1P8 11001493 Ki = 39810.72 nM T16347 CT4H0O 11006141 IC50 = 5300 nM T16347 C78GFD 11020078 Ki = 2500 nM T16347 C8YV9L 11034520 Ki = 6025.6 nM T16347 CWZ2F6 11036155 Ki = 12000 nM T16347 C2U4EM 11038621 Ki = 9100 nM T16347 CVSN28 11044461 Ki = 250000 nM T16347 C16WZS 11045948 IC50 = 230000 nM T16347 CH3Z0K 11046051 Ki = 74000 nM T16347 C7C2SQ 11047141 Ki = 9000 nM T16347 CGP3V2 11057341 Ki = 11000 nM T16347 C6L9JY 11061339 Ki = 370 nM T16347 CAC81E 11064049 Ki = 1096478.2 nM T16347 CU8DA1 11069603 Ki = 42000 nM T16347 CI86XU 11069872 IC50 > 50000 nM T16347 CTCQ74 11092597 Ki = 14000 nM T16347 CSQP94 11093509 Ki = 31.62 nM T16347 CC1E9B 11100844 Ki = 8700 nM T16347 COLP53 11109453 Ki = 5100 nM T16347 C4LRH3 11111298 Ki = 2500 nM T16347 C6RJW1 11115025 Ki = 12.59 nM T16347 C1R2EU 11115308 Ki = 390 nM T16347 C7J1PF 11117661 Ki = 1698243.65 nM T16347 CV9KN6 11119535 IC50 = 9400000 nM T16347 CCU95R 11131230 Ki = 35000 nM T16347 CZ9A1P 11136043 Ki = 130 nM T16347 CV1T6U 11138143 IC50 = 3300000 nM T16347 CAS59E 11139219 IC50 = 790000 nM T16347 C03TXN 11155758 IC50 = 51400 nM T16347 CAB53D 11177475 IC50 = 14800 nM T16347 C7U1BT 11186786 IC50 = 20700 nM T16347 CDOU70 11187348 IC50 > 30000 nM T16347 CCOP61 11189464 Ki = 50118.72 nM T16347 C6MH4V 11199403 IC50 = 19800 nM T16347 CNW19H 11213350 IC50 = 23600 nM T16347 CL81UD 11226572 IC50 = 35 nM T16347 C1SPI9 11236319 IC50 = 101100 nM T16347 CO1DS6 11236561 IC50 = 120200 nM T16347 C8AD0Y 11266347 Ki = 45000 nM T16347 COF17B 11268298 IC50 = 8600 nM T16347 CFW5X8 11282472 IC50 = 26000 nM T16347 CVS8I5 11302670 IC50 = 3.97 ug.mL-1 T16347 C37CAG 11316438 IC50 = 82100 nM T16347 C8R5SD 11316815 IC50 = 242000 nM T16347 COLN21 11327911 IC50 = 198000 nM T16347 C2WP1J 11343454 IC50 = 2500 nM T16347 CQFG80 11346860 Ki = 30000 nM T16347 C46UEQ 11346984 IC50 = 128800 nM T16347 CLMG62 11362207 Ki = 50118.72 nM T16347 CK01AH 11381519 IC50 = 15400 nM T16347 CZWS86 11382597 IC50 = 11700 nM T16347 CFYE08 11390413 IC50 > 45000 nM T16347 CR5A7F 11392873 IC50 > 32000 nM T16347 C4CHS5 11431694 IC50 = 224800 nM T16347 CRO73E 11432549 IC50 > 200000 nM T16347 COIR53 11456678 Ki = 740 nM T16347 C0X2AF 11462303 IC50 = 18300 nM T16347 C9O7LT 11497557 IC50 = 600 nM T16347 C81ECX 11513780 IC50 = 17500 nM T16347 CRPL64 11516963 IC50 = 800 nM T16347 C5G0SI 11569279 IC50 = 2999162.52 nM T16347 CJ0B6K 11596309 IC50 = 310 nM T16347 CJ36ZF 11619012 IC50 = 4850 nM T16347 C0YF1L 11633740 Ki = 3100 nM T16347 C5AM4Q 11669443 IC50 = 100000000 nM T16347 CX4E6H 11671705 IC50 = 600 nM T16347 C8V9FL 11678073 IC50 = 85100 nM T16347 CP4JE6 11684950 IC50 = 220 nM T16347 CV4D5H 11691610 IC50 = 16000 nM T16347 COBH46 11693218 IC50 = 35 nM T16347 COH8T4 11699721 IC50 = 590 nM T16347 C3P1EW 11702273 Ki = 4100 nM T16347 C80EXT 11711911 IC50 = 100000000 nM T16347 C9LUE3 11720639 IC50 = 940 nM T16347 CVY25D 11723433 IC50 = 10400 nM T16347 C6H9EC 11729429 IC50 = 3800000 nM T16347 CEN6B1 11733586 Ki = 9772.37 nM T16347 CPTU86 11745998 Ki = 75000 nM T16347 CS1C6R 11746409 Ki = 1995262.31 nM T16347 C2VEB7 11753144 IC50 = 8610 nM T16347 CL9QN7 11757194 IC50 < 10000 nM T16347 CC5MI6 11770718 IC50 = 9400000 nM T16347 C26NZK 11776892 IC50 = 35700 nM T16347 C6A1LM 11786814 Ki = 4 nM T16347 CH09LO 11790598 IC50 > 3200000 nM T16347 CTR50I 11799727 IC50 = 1300 nM T16347 C8RHW3 11800217 IC50 = 346.74 nM T16347 CU62IW 11800547 IC50 = 410 nM T16347 C25XGH 11801834 IC50 = 850 nM T16347 CN8SR4 11802196 IC50 = 178 nM T16347 C5DP0W 11808397 Ki = 900000 nM T16347 C84QMT 11809534 Ki = 10000 nM T16347 CL3B8H 11813772 Ki = 2000 nM T16347 CV1ZX3 11814026 Ki = 9000 nM T16347 COZR52 11824758 Ki = 14000 nM T16347 CK2L6A 11824932 Ki = 24000 nM T16347 COLQ31 11826482 Ki = 8000 nM T16347 CW0Y1T 11826936 Ki = 15000 nM T16347 C1G4MV 11827337 Ki = 1200 nM T16347 C6SM1U 11828719 Ki = 560 nM T16347 CF17EN 11840289 IC50 = 2100 nM T16347 CM1XL8 11844603 IC50 > 100000 nM T16347 C75UVA 11844604 IC50 > 100000 nM T16347 C03MRZ 11869658 IC50 = 5050 nM T16347 CTM3Y4 11948628 Ki = 30000 nM T16347 C1SLO0 11948629 Ki = 32000 nM T16347 CEQ0N5 11995580 IC50 = 21200 nM T16347 C5OG6C 11995581 IC50 > 60000 nM T16347 C36LEV 12001105 IC50 = 200 nM T16347 CU52BJ 12051847 IC50 = 7800 nM T16347 C4XF5D 12069327 IC50 = 23900 nM T16347 C6DK4E 12070920 IC50 = 560 nM T16347 CRC5K3 12094720 IC50 = 16200 nM T16347 C9DTX2 12098451 IC50 = 21600 nM T16347 CV7E4B 12109536 IC50 = 29000 nM T16347 CEFU08 12109538 IC50 = 24000 nM T16347 CBXM15 12109539 IC50 = 24000 nM T16347 C9AHN6 12142457 IC50 = 29000 nM T16347 CN6QI5 12299984 IC50 = 16790 nM T16347 C4DQ9P 12302281 IC50 = 8930 nM T16347 CL06YJ 12302571 IC50 > 30000 nM T16347 CKNP83 12309637 IC50 = 18690 nM T16347 CB6Q3O 12315075 IC50 = 20100 nM T16347 C4Q5AX 12458245 IC50 > 60000 nM T16347 C8SB0U 12585551 IC50 = 640000 nM T16347 CPV08O 12658768 IC50 > 20000 nM T16347 CG73WI 12773960 Ki = 200 nM T16347 C9H3UP 12968370 IC50 = 10000 nM T16347 CY2S7W 12968371 IC50 = 1500000 nM T16347 CX27OP 12968372 IC50 = 430000 nM T16347 CZEV28 12968373 IC50 = 3700000 nM T16347 C1GK0W 12968374 IC50 = 2500000 nM T16347 C3ALV1 12968375 IC50 = 650000 nM T16347 CW3A8Q 12968376 IC50 = 13000000 nM T16347 CW61YC 12968377 IC50 = 4400000 nM T16347 C8ZUE9 12968378 IC50 = 5300000 nM T16347 C0OP4N 12968379 IC50 = 4600000 nM T16347 CGAK08 13210058 Ki = 3162277.66 nM T16347 C68QTW 13241303 IC50 = 7980 nM T16347 CW7Z8X 13441995 IC50 = 1420 nM T16347 C9LH2Z 13545019 IC50 = 5050 nM T16347 CE8Y4G 13779016 IC50 = 360200 nM T16347 C7KY9W 13857523 IC50 > 30000 nM T16347 C4SNP7 13915902 IC50 = 13210 nM T16347 CPG7W6 13922429 IC50 = 403000 nM T16347 C8ZB9F 13922432 IC50 = 148000 nM T16347 CA19MJ 13965473 IC50 = 70000 nM T16347 CUD2T6 13994560 IC50 = 14700 nM T16347 CO4Y6W 14017299 IC50 > 30000 nM T16347 C4KW7G 14024697 IC50 > 120000 nM T16347 CT60GS 14136878 IC50 > 30000 nM T16347 C8D1IK 14136881 IC50 = 7400 nM T16347 C5C4SD 14161396 IC50 = 10340 nM T16347 CK4AC9 14161397 IC50 = 41700 nM T16347 CW08FH 14208454 IC50 = 2610 nM T16347 C5XQH1 14237659 IC50 = 500 nM T16347 CW6K1I 14309760 IC50 = 1030 nM T16347 CB08WX 14334313 IC50 = 1940 nM T16347 CPX02C 14336535 IC50 >= 20 ug.mL-1 T16347 CZK16N 14539883 IC50 > 80000 nM T16347 CQYM59 14550005 IC50 > 4000000 nM T16347 C0TGO3 14564364 IC50 = 9000 nM T16347 CRDX95 14564373 IC50 = 21200 nM T16347 C3ZN1P 14602300 IC50 > 200000 nM T16347 CBNE97 14658766 IC50 = 18000 nM T16347 C2BC5F 14753570 IC50 = 15300 nM T16347 C63EZQ 14785818 IC50 = 78000 nM T16347 C18JXA 15233562 IC50 = 64900 nM T16347 CW7IE0 15273394 IC50 = 5730 nM T16347 C78CIE 15273395 IC50 = 440 nM T16347 CH3BG7 15292820 IC50 = 85500 nM T16347 CDJP28 15322751 IC50 = 1130 nM T16347 CU13IF 15384192 IC50 = 1200000 nM T16347 C7Z0AJ 15384193 IC50 = 800000 nM T16347 C57EUC 15384194 Ki = 3600 nM T16347 CVKT94 15429542 IC50 = 49970 nM T16347 C7QJO4 15479638 IC50 = 2600 nM T16347 CRH5W9 15485891 IC50 = 60 nM T16347 CKPF01 15485898 IC50 = 89 nM T16347 C6KN1Z 15486039 IC50 = 386000 nM T16347 CPG80C 15486040 IC50 = 167100 nM T16347 CCQ23W 15486041 IC50 = 88700 nM T16347 C4RZO6 15486042 IC50 = 57900 nM T16347 CYR0I9 15520072 Ki = 61000 nM T16347 CI9RD5 15588112 Ki > 1000000 nM T16347 C1Z2UC 15588116 Ki = 18000 nM T16347 CRX7T8 15588121 IC50 > 2500000 nM T16347 CQA34E 15664151 IC50 = 400 nM T16347 C42ABS 15719494 IC50 = 17400 nM T16347 C9LXO3 15742118 IC50 = 32600 nM T16347 C3PJT1 15818599 IC50 = 4500 nM T16347 C4BP6X 15859320 IC50 = 22700 nM T16347 CI2PE0 15981925 IC50 = 560 nM T16347 CIE95V 15981929 IC50 = 350 nM T16347 CI7SD3 15982441 IC50 = 1850 nM T16347 CO4R1J 15982447 IC50 = 270 nM T16347 C36FCN 15982567 IC50 = 1370 nM T16347 CMH24O 15982706 IC50 = 530 nM T16347 C7R2AB 15982964 IC50 = 1660 nM T16347 C17FHP 15982965 IC50 = 480 nM T16347 CT7O6A 15982966 IC50 = 510 nM T16347 C9C8FP 15982968 IC50 = 260 nM T16347 CM42PV 15983098 IC50 = 250 nM T16347 CFZ0J8 15983472 IC50 = 1160 nM T16347 C7KD9X 15983473 IC50 = 2790 nM T16347 CE03OL 15983474 IC50 = 500 nM T16347 CW47VB 15983717 IC50 = 1000 nM T16347 C35KBS 15983725 IC50 = 610 nM T16347 CL81AH 15983850 IC50 = 2390 nM T16347 CFP7G3 15983852 IC50 = 1340 nM T16347 CTD4R1 15983861 IC50 = 1150 nM T16347 C2PJ5U 16036807 Ki = 13 nM T16347 CGQ81X 16046117 Ki = 140 nM T16347 CQY9A2 16058638 Ki = 300 nM T16347 C9GNW0 16086577 IC50 > 10 ug.mL-1 T16347 C1G6XV 16091635 IC50 = 6330 nM T16347 CRY60F 16104905 IC50 > 80000 nM T16347 CYH52T 16109844 IC50 = 3.1 ug.mL-1 T16347 CLJ61H 16109845 IC50 > 10000 nM T16347 C72XGN 16121783 IC50 = 14760 nM T16347 C0P4TQ 16220825 IC50 > 1000000 nM T16347 C17KIT 16220826 IC50 > 1000000 nM T16347 C0XZV4 16220827 IC50 = 1000000 nM T16347 CMX13P 16221752 IC50 > 1000000 nM T16347 C2PT9M 16221754 IC50 > 1000000 nM T16347 CM65WP 16221756 IC50 > 1000000 nM T16347 CY83SR 16221757 IC50 = 24000 nM T16347 C2PEO3 16634009 IC50 = 9000 nM T16347 C4M1AU 16659198 IC50 = 230 nM T16347 C8W2YO 16664188 Ki = 3000 nM T16347 C5O4NE 16737096 IC50 = 18900 nM T16347 CSJ3D6 16737249 IC50 > 60000 nM T16347 C4VB7R 16738021 IC50 = 16500 nM T16347 CES7C6 17403725 IC50 = 44000 nM T16347 C5K9MX 17748269 Ki = 9400 nM T16347 CY5F3K 17757503 IC50 = 80 nM T16347 C34HXV 17758005 Ki = 390 nM T16347 C8SF4H 17758007 Ki = 310 nM T16347 C8QR7X 17758127 Ki = 190 nM T16347 C0XO5C 17758128 Ki = 300 nM T16347 CHN9Z0 17758226 Ki = 44 nM T16347 CJ0QS5 17758343 Ki = 8 nM T16347 C02TBQ 17758453 Ki = 74 nM T16347 CGF7A8 17758455 Ki = 310 nM T16347 C5VMH8 17758565 Ki = 13 nM T16347 C2HML5 17758567 Ki = 10 nM T16347 CYQH72 17758677 Ki = 6 nM T16347 C6T4JF 17758679 Ki = 6 nM T16347 CGH9S1 17758681 Ki = 2 nM T16347 C8O1LY 17758809 Ki = 14 nM T16347 C2RLY7 17758810 Ki = 4 nM T16347 CDY87I 17758812 Ki = 3 nM T16347 CF34ND 17758916 Ki = 3 nM T16347 CLWK36 17758917 Ki = 1000 nM T16347 C8R3JV 17758918 Ki = 2000 nM T16347 CFS4L8 17758919 Ki = 2000 nM T16347 C6D3LQ 17758920 Ki = 470 nM T16347 C6HU1X 17758921 Ki = 200 nM T16347 CMP0U6 17758922 Ki = 120 nM T16347 C94LBM 17759043 Ki = 26 nM T16347 C2ZPI7 17759044 Ki = 3800 nM T16347 C1PG3M 17759045 Ki = 390 nM T16347 C7OTA4 17759046 Ki = 55 nM T16347 CDG4T0 17759047 Ki = 2000 nM T16347 CA3TS5 17759048 Ki = 0.68 nM T16347 CV7WM8 17759187 Ki = 24 nM T16347 C6V4LO 17759188 Ki = 7 nM T16347 CLH5A0 17759189 Ki = 38 nM T16347 CNKU76 17759190 Ki = 5 nM T16347 CD79PM 17759191 Ki = 4 nM T16347 C9JT7Y 17759313 Ki = 2 nM T16347 CH5Q1X 17759314 Ki = 1 nM T16347 CYW2B5 17759315 Ki = 3 nM T16347 C1LKX3 17759664 Ki = 1700 nM T16347 C0US9T 17759666 Ki = 4000 nM T16347 CZV56K 17759775 Ki = 2100 nM T16347 C1QP2U 17759776 Ki = 2100 nM T16347 C5B2XE 17759777 Ki = 440 nM T16347 CQ1VG3 17759778 Ki = 680 nM T16347 CX1N0F 17759780 Ki = 210 nM T16347 CW0A2H 17777098 Ki = 2500000 nM T16347 C2Y4MT 18003344 IC50 = 21000 nM T16347 CD8Q6T 18006434 IC50 = 4800 nM T16347 C1QXG6 18178937 IC50 = 12900 nM T16347 C9O8GW 18185289 IC50 = 2500 nM T16347 C5TE6K 18398682 IC50 = 8040 nM T16347 CBQO20 18398709 IC50 = 2000 nM T16347 C1E8HM 18476765 Ki = 6500 nM T16347 CN9EH2 18864297 IC50 = 10000 nM T16347 C6ZEL2 18864298 IC50 = 85000 nM T16347 CF24QL 18864314 IC50 = 4600 nM T16347 CBJ60K 18864315 IC50 = 1600 nM T16347 CJ4P9E 18957696 IC50 > 500000 nM T16347 C3TV7F 19779154 IC50 = 65000 nM T16347 C37LQG 19880831 IC50 = 57000 nM T16347 C68VHP 21121150 IC50 = 9500 nM T16347 CG2W8S 21145050 IC50 = 17580 nM T16347 C12GAZ 21145366 Ki = 3200 nM T16347 CFBX76 21145371 IC50 = 7 nM T16347 C09VUC 21145380 Ki = 7943.28 nM T16347 CRXU06 21148065 IC50 = 2400 nM T16347 CKNX31 21213049 IC50 = 122000 nM T16347 CH91UW 21265708 IC50 = 800 nM T16347 CLI13Y 21265715 IC50 = 60 nM T16347 C40CYN 21265722 IC50 = 390 nM T16347 CQ6H5V 21585575 IC50 = 7470 nM T16347 C7BM3L 21591148 IC50 = 3000 nM T16347 CU8W6F 21591394 IC50 = 215000 nM T16347 CP4BL9 21594119 IC50 = 6800 nM T16347 C3T9AB 21594122 Ki = 3100 nM T16347 C9DQ4F 21721847 IC50 = 4310 nM T16347 CTKW85 21770907 Ki = 18390 nM T16347 CLJ16A 21773091 IC50 = 11.6 ug.mL-1 T16347 C54IUM 21778115 IC50 = 680 nM T16347 CA27DS 21778221 IC50 >= 20 ug.mL-1 T16347 CEO71J 21778335 IC50 = 6.8 ug.mL-1 T16347 C8VI1J 21878530 IC50 = 80 nM T16347 C4HZL2 21878534 IC50 = 160 nM T16347 C2W9PG 21878588 IC50 = 67 nM T16347 C18NUG 21878691 IC50 = 110 nM T16347 CD39RP 21878699 IC50 = 80 nM T16347 CO41ZD 21878897 IC50 = 80 nM T16347 CB16YQ 21878911 IC50 = 170 nM T16347 CT69OF 21878965 IC50 = 130 nM T16347 C0J5HQ 21878987 IC50 = 94 nM T16347 CF08UN 21879012 IC50 = 45 nM T16347 C34YDM 21879031 IC50 = 60 nM T16347 CG3R2M 21879040 IC50 = 51 nM T16347 CT5PL3 21879063 IC50 = 48 nM T16347 C1SLD6 21879071 IC50 = 160 nM T16347 CHE7G6 21879098 IC50 = 240 nM T16347 CH0I7R 21879153 IC50 = 63 nM T16347 CD20GT 21879220 IC50 = 85 nM T16347 CJ92HM 21879229 IC50 = 460 nM T16347 CK6UZ2 21879268 IC50 = 120 nM T16347 C5WO3N 21879347 IC50 = 160 nM T16347 CCUY37 21879425 IC50 = 43 nM T16347 C5R3DM 21879462 IC50 = 300 nM T16347 C1HK7X 21879487 IC50 = 77 nM T16347 C56YWT 21879558 IC50 = 110 nM T16347 C1OR3D 22084082 Ki = 18000 nM T16347 C18FPX 22256263 IC50 = 1180000 nM T16347 CHG9X6 22271909 Ki = 251.19 nM T16347 CCZQ38 22280049 IC50 = 20000 nM T16347 CI7Y1R 22327692 IC50 = 2150 nM T16347 CA5BH7 23090222 IC50 = 20000 nM T16347 C2E1ZQ 23423270 Ki = 3300000 nM T16347 C8CM6X 23427285 IC50 = 15000 nM T16347 CP61IS 23624833 IC50 >= 20 ug.mL-1 T16347 CCL5Q6 23644688 Ki = 3400 nM T16347 CIF58J 23644689 Ki = 1300 nM T16347 CC32QO 23644690 Ki = 125.89 nM T16347 C7R8ES 23644691 Ki = 430 nM T16347 C5WR6S 23644692 Ki = 199.53 nM T16347 C0VJ6H 23644693 Ki = 710 nM T16347 CJT9A0 23644694 Ki = 100 nM T16347 CL1F3M 23644695 Ki = 398.11 nM T16347 CK81YQ 23644696 Ki = 1700 nM T16347 C9FLE4 23646398 IC50 > 500000 nM T16347 CR1D8X 23646399 IC50 = 19000 nM T16347 C6TPG0 23646400 IC50 = 16700 nM T16347 CCNB08 23646401 IC50 = 8230 nM T16347 CYXL64 23646402 IC50 = 183700 nM T16347 CIO93Z 23646403 IC50 = 146000 nM T16347 CCD0J5 23646404 IC50 = 93400 nM T16347 CUH19M 23646468 Ki = 250 nM T16347 C4BS8C 23646469 Ki = 5000 nM T16347 C7UDP0 23646520 IC50 = 660693.45 nM T16347 C8QN5P 23646521 IC50 = 149968.48 nM T16347 CR6X9Y 23646522 IC50 = 49 nM T16347 C9AI3W 23646523 IC50 = 163 nM T16347 CDIV60 23646551 Ki = 125.89 nM T16347 CRC68Q 23646552 Ki = 540 nM T16347 C2WM9P 23646560 Ki = 8800 nM T16347 CX0Q1J 23646561 Ki = 6100 nM T16347 C0A1IJ 23646566 Ki > 200000 nM T16347 CPZB65 23646567 Ki > 200000 nM T16347 CI1CA2 23646568 Ki > 200000 nM T16347 CC7W8Z 23646569 Ki = 218776.16 nM T16347 CDN7K5 23646574 Ki = 12589.25 nM T16347 CZU27A 23646660 Ki > 1000000 nM T16347 C8BSV1 23646661 Ki > 1000000 nM T16347 C8PY9K 23646662 Ki = 1400 nM T16347 CBLI14 23646663 Ki = 4000 nM T16347 CW29HQ 23646664 Ki = 3300 nM T16347 CIVL25 23646665 Ki = 5000 nM T16347 C3B8HZ 23646666 Ki = 3000 nM T16347 CWGH80 23646667 Ki = 570 nM T16347 CQ2HS8 23646668 Ki = 1600 nM T16347 C6NH3C 23646669 Ki = 1000 nM T16347 CXCF89 23646670 Ki = 500 nM T16347 CPR47T 23646671 Ki = 620 nM T16347 C7ER2Q 23646672 Ki = 680 nM T16347 C4ZS8H 23646673 Ki = 600 nM T16347 CT04KC 23646674 Ki = 2500 nM T16347 CM84CI 23646675 Ki = 740 nM T16347 CCMG59 23646676 Ki = 200 nM T16347 CV9LN8 23646677 Ki = 1200 nM T16347 C0M8WR 23646678 Ki = 1000 nM T16347 CRB0J9 23646679 Ki = 360 nM T16347 CV48EU 23646680 Ki = 250 nM T16347 CU8BR2 23646681 IC50 = 480 nM T16347 CGL09B 23646682 IC50 > 10000 nM T16347 CI29QS 23646683 IC50 = 330 nM T16347 C60DXK 23646684 IC50 = 1300 nM T16347 C1XFN4 23646685 IC50 = 740 nM T16347 CG3ZX8 23646686 IC50 = 490 nM T16347 C2K6EF 23646687 IC50 = 420 nM T16347 C90STC 23646688 IC50 = 660 nM T16347 CQ9IT6 23646689 IC50 = 440 nM T16347 C0L2OB 23646690 IC50 = 970 nM T16347 CQ28SK 23646691 IC50 = 2400 nM T16347 C8X2LC 23646692 IC50 = 350 nM T16347 CIF67N 23646693 IC50 = 550 nM T16347 CCL50B 23646694 IC50 = 470 nM T16347 CHX9R7 23646695 IC50 = 1100 nM T16347 CT0BY3 23646696 IC50 = 500 nM T16347 C8C4WG 23646697 IC50 = 620 nM T16347 C21CIR 23646698 IC50 = 1100 nM T16347 CN2HS0 23646699 IC50 = 150 nM T16347 C5MB9Z 23646700 IC50 = 410 nM T16347 CBU1P9 23646701 IC50 = 470 nM T16347 C37DIZ 23646702 IC50 = 280 nM T16347 CK6DV9 23646703 IC50 = 1600 nM T16347 C3L9WM 23646704 IC50 = 400 nM T16347 C9FCT2 23646705 IC50 = 460 nM T16347 C9P2YI 23647189 Ki = 540 nM T16347 CT2Y6O 23647190 Ki = 1200 nM T16347 C9W0AH 23647191 Ki = 4700 nM T16347 CIT62P 23647192 Ki = 2500 nM T16347 CD7Z1Q 23655080 IC50 = 13600 nM T16347 C9ZT7V 23661682 IC50 = 14900 nM T16347 CM1G4E 23673589 Ki = 49000 nM T16347 C0V4TI 23675509 Ki = 98000 nM T16347 C39BLE 23702953 IC50 = 230000 nM T16347 CVQU13 23705237 IC50 = 35 nM T16347 C72BMW 23843929 IC50 = 2540 nM T16347 CE7IG6 24073040 IC50 = 12000 nM T16347 CF9O0N 24178900 IC50 = 3710 nM T16347 C8XWY9 24178901 IC50 = 1700 nM T16347 CDTE90 24180456 Ki = 1100 nM T16347 C21ECL 24180507 Ki = 6500 nM T16347 C5O0SV 24204784 IC50 > 100000 nM T16347 CUYA53 24206831 Ki = 7900 nM T16347 CB06SX 24206834 Ki = 7900 nM T16347 C7NBT0 24243261 IC50 = 9390 nM T16347 CZL2T6 24815971 IC50 = 70 nM T16347 CP53VK 24834047 IC50 = 35100 nM T16347 CS18TW 24857885 IC50 = 120 nM T16347 CS8M7X 24861961 IC50 = 23200 nM T16347 CYV30B 24873529 IC50 = 3000 nM T16347 C3IE8L 24936165 IC50 = 32 nM T16347 CSB53M 24939957 IC50 > 24400 nM T16347 CN82VP 25010727 IC50 = 1400 nM T16347 CSPH15 25012043 IC50 > 36000 nM T16347 CEC8V2 25012694 IC50 = 17890 nM T16347 C9I4NZ 25013669 IC50 = 14690 nM T16347 C7IB6G 25013826 IC50 = 10890 nM T16347 C5R1CK 25013830 IC50 = 18020 nM T16347 CY4AB6 25013832 IC50 = 19850 nM T16347 CBJK01 25014012 IC50 = 9540 nM T16347 C6OWQ0 25014013 IC50 = 8920 nM T16347 CIV15S 25014015 IC50 = 9440 nM T16347 CH8UE7 25014220 IC50 = 8440 nM T16347 CA4RK0 25014221 IC50 = 13460 nM T16347 CE9B6H 25014222 IC50 = 9320 nM T16347 CJWZ03 25014223 IC50 = 19020 nM T16347 CJCY62 25055680 IC50 = 60 nM T16347 CLS6X2 25055681 IC50 = 250 nM T16347 CWMV64 25056374 IC50 = 330 nM T16347 CNS2U7 25056375 IC50 = 90 nM T16347 CU59JO 25056378 IC50 = 310 nM T16347 C9BET0 25056379 IC50 = 1260 nM T16347 CT0H3U 25056635 IC50 = 14000 nM T16347 CC2Q6Z 25056895 IC50 = 45 nM T16347 CE8J2D 25056896 IC50 = 27 nM T16347 CF6AD0 25101398 IC50 = 153000 nM T16347 C8SB5R 25101399 IC50 = 84000 nM T16347 CJ9E8P 25101400 IC50 = 91000 nM T16347 C1Y0KM 25101546 Ki = 6300 nM T16347 CVNR04 25101547 IC50 = 39000 nM T16347 C3KQ1I 25101548 IC50 = 67000 nM T16347 CJHV56 25101549 IC50 = 27000 nM T16347 CX93QV 25102798 IC50 < 30 nM T16347 C6CEZ5 25103887 IC50 = 125 nM T16347 CN7HW4 25136079 IC50 > 30000 nM T16347 CZ4M3C 25141412 IC50 = 3000 nM T16347 CL9T6N 25147600 IC50 = 17900 nM T16347 C7TJ9A 25147601 IC50 = 18200 nM T16347 CA04MU 25154757 IC50 = 770 nM T16347 CN5PH6 25198918 IC50 = 4550 nM T16347 CZY40D 25198919 IC50 = 1860 nM T16347 CX5UE4 25199063 IC50 = 3500 nM T16347 CHA3V1 25199065 IC50 = 3360 nM T16347 CC0RP7 25199068 IC50 = 3510 nM T16347 C5I6ZY 25199187 IC50 = 5700 nM T16347 CQ6YS4 25199188 IC50 = 2500 nM T16347 C3R1OG 25208124 IC50 > 80000 nM T16347 CP9K1X 25211684 IC50 = 39500 nM T16347 C09KZA 25262525 IC50 = 11800 nM T16347 C4WM9S 25262527 IC50 = 14300 nM T16347 C4QA6B 25761582 IC50 = 679000 nM T16347 CFVH68 25761598 IC50 = 24560 nM T16347 C1HT4Y 25795027 IC50 = 14000 nM T16347 CP6I9Y 29248068 IC50 = 68000 nM T16347 CXN2V1 29920877 IC50 = 10000 nM T16347 C17OYW 38361391 IC50 = 17400 nM T16347 CZL19R 39834448 IC50 > 100000 nM T16347 CEY7Z2 40557055 IC50 > 20000 nM T16347 C5CT1N 42607541 IC50 = 5000 nM T16347 C3P8XN 42644186 IC50 = 1790 nM T16347 C98IOF 42644187 IC50 = 1430 nM T16347 CSH73Q 43230121 IC50 = 1000 nM T16347 C07SPI 44138095 IC50 = 58000 nM T16347 CNJ94H 44138096 IC50 = 86000 nM T16347 COZ1C5 44138908 IC50 = 35400 nM T16347 CFP1I4 44138909 IC50 = 27200 nM T16347 CJV2U5 44139659 IC50 = 429 nM T16347 CJF79U 44139660 IC50 = 383.7 nM T16347 CEJ6U5 44139661 IC50 = 553.3 nM T16347 CN72DB 44139662 IC50 = 510.3 nM T16347 C59BUM 44139779 IC50 = 385.7 nM T16347 CDV3R8 44139780 IC50 = 353.7 nM T16347 CV4X7D 44139781 IC50 = 164.7 nM T16347 CY9LW6 44139782 IC50 = 135.7 nM T16347 CJ01NF 44139783 IC50 = 668.7 nM T16347 CJQU21 44139784 IC50 = 637.7 nM T16347 CQK73G 44139926 IC50 = 104.3 nM T16347 CEC01T 44139927 IC50 = 95.67 nM T16347 C34VTJ 44139928 IC50 = 80 nM T16347 CHSY93 44139930 IC50 = 2897 nM T16347 C0F5RG 44139931 IC50 = 2753 nM T16347 CZA86R 44139932 IC50 = 167.3 nM T16347 C8H6VX 44140057 IC50 = 114.3 nM T16347 CXT39E 44140058 IC50 = 566.7 nM T16347 C8L0PD 44140061 IC50 = 304 nM T16347 CB21AP 44140190 IC50 = 148.7 nM T16347 CYW23M 44140191 IC50 = 373.7 nM T16347 CR7WY9 44140317 IC50 = 518.7 nM T16347 C6QO0X 44140445 IC50 = 113 nM T16347 CNDB57 44140446 IC50 = 358.3 nM T16347 CL04IU 44156271 IC50 = 14000 nM T16347 C6JEK3 44156972 IC50 = 7700 nM T16347 CTCI39 44156973 IC50 = 1000 nM T16347 CNY45K 44178673 IC50 > 30000 nM T16347 C2ITW9 44188089 IC50 = 6860 nM T16347 CWT3E1 44188090 IC50 = 1500 nM T16347 C4I7WB 44218137 IC50 = 240 nM T16347 C4KO9Y 44265540 IC50 = 940 nM T16347 C73QKU 44265541 IC50 = 90 nM T16347 CJ6HG2 44265546 IC50 = 360 nM T16347 CF2L9H 44265570 IC50 = 16000 nM T16347 CJ5C0R 44265576 IC50 = 160 nM T16347 CK1Q2C 44265649 IC50 = 110 nM T16347 COD4L3 44265670 IC50 = 32 nM T16347 CWTQ56 44265697 IC50 = 20 nM T16347 C8D9TY 44265698 IC50 = 88 nM T16347 CB1H0Y 44265797 IC50 = 240 nM T16347 CNLW94 44265857 IC50 = 74 nM T16347 C7JLB1 44265863 IC50 = 98 nM T16347 CD79RG 44265874 IC50 = 46 nM T16347 CJQE06 44265877 IC50 = 16 nM T16347 CSM7R2 44265887 IC50 = 19 nM T16347 C69UNK 44274769 IC50 = 460 nM T16347 C3GZP5 44285457 IC50 = 179 nM T16347 C1L3HZ 44291989 IC50 = 4820 nM T16347 C8IPW4 44292106 IC50 = 4710 nM T16347 C5T8GM 44292122 IC50 = 2960 nM T16347 CVR30X 44300873 IC50 = 320000 nM T16347 CJDG23 44300940 IC50 = 1340 nM T16347 C03NFT 44300941 IC50 = 2250 nM T16347 C81TAY 44300976 IC50 = 1600 nM T16347 CN5X7V 44300978 IC50 = 1070 nM T16347 CO0ZJ4 44300994 IC50 = 650 nM T16347 CB5Y3T 44301003 IC50 = 2040 nM T16347 C5QE9K 44301004 IC50 = 920 nM T16347 CPH9S3 44301018 IC50 = 2690 nM T16347 C7N5XS 44301035 IC50 = 2300000 nM T16347 CZHC76 44301073 IC50 = 5400 nM T16347 C18XNS 44301074 IC50 = 4200 nM T16347 CQF18L 44301080 IC50 = 940 nM T16347 C7DK9B 44301081 IC50 = 680 nM T16347 CX7U5B 44301087 IC50 = 650 nM T16347 CQY28R 44301093 IC50 = 3300 nM T16347 C5K3US 44301125 IC50 = 5240 nM T16347 C74BFI 44301128 IC50 = 430 nM T16347 CDJ1S7 44301133 IC50 = 1540 nM T16347 CXG2V5 44301137 IC50 = 920 nM T16347 CJZ79P 44301148 IC50 = 2150 nM T16347 CP7LO1 44301154 IC50 = 500 nM T16347 C3SA4Y 44301171 IC50 = 36470 nM T16347 CUK41J 44301182 IC50 = 610 nM T16347 CSQ4G2 44301245 IC50 = 330 nM T16347 CL0G7R 44301247 IC50 = 1010 nM T16347 C7BN9L 44301259 IC50 = 270 nM T16347 CF32KE 44301278 IC50 = 2070 nM T16347 CBTX21 44301279 IC50 = 2540 nM T16347 CE72AG 44301347 IC50 = 1170 nM T16347 CA1L9K 44301367 IC50 = 1010 nM T16347 C5C0RK 44301368 IC50 = 1540 nM T16347 C96YVT 44301380 IC50 = 4560 nM T16347 CJZ34O 44301381 IC50 = 3000 nM T16347 C2TV9N 44303254 IC50 > 360000 nM T16347 CK78HD 44303432 IC50 = 21000 nM T16347 C1X8YT 44303433 IC50 = 160000 nM T16347 CPC2M1 44303451 IC50 = 87000 nM T16347 CZ5MD3 44303453 IC50 = 68000 nM T16347 CT2HK6 44303463 IC50 = 50000 nM T16347 CN89QP 44303489 IC50 > 100000 nM T16347 C7E4AP 44303513 IC50 = 4400 nM T16347 C5H0VL 44303516 IC50 > 320000 nM T16347 C5Y6QE 44303518 IC50 > 100000 nM T16347 C7GJ6P 44303523 IC50 = 185000 nM T16347 CHK98F 44303528 IC50 = 40500 nM T16347 CBI8O6 44303580 IC50 = 110000 nM T16347 C0X8JR 44303638 IC50 > 310000 nM T16347 CXN80T 44303639 IC50 > 290000 nM T16347 CZTE47 44303667 IC50 = 5400 nM T16347 CYL2E5 44303668 IC50 = 17000 nM T16347 CIT1K3 44303684 IC50 > 100000 nM T16347 CMPA04 44303685 IC50 > 100000 nM T16347 CF6XD7 44306264 Ki = 9100 nM T16347 CE5AT9 44306295 Ki = 9800 nM T16347 CWM2U3 44306738 Ki = 17300 nM T16347 CL7J8V 44306768 Ki > 100000 nM T16347 CON29A 44310730 IC50 = 21500 nM T16347 CV0AM3 44311047 IC50 = 9000 nM T16347 CBGU12 44320386 Ki = 29000 nM T16347 CMRN52 44320416 IC50 = 3100 nM T16347 CXY53I 44320455 IC50 = 54700 nM T16347 C1QUS4 44320456 IC50 = 116000 nM T16347 CAN5I3 44320598 IC50 = 700 nM T16347 CB98UX 44320599 IC50 = 1500 nM T16347 C9TQJ8 44320600 IC50 = 700 nM T16347 C9B7NR 44320648 IC50 = 8300 nM T16347 C3M4BJ 44320663 IC50 = 19400 nM T16347 CZB2P4 44320672 IC50 = 44000 nM T16347 C8AY6U 44320673 IC50 = 800 nM T16347 CGT4B1 44320854 IC50 = 1400 nM T16347 C3OH9T 44320855 IC50 = 4000 nM T16347 C7O9ND 44320874 IC50 = 1410 nM T16347 C4GN9S 44320886 IC50 = 72000 nM T16347 C94YNR 44329391 Ki = 12000 nM T16347 CT27EC 44329513 IC50 = 29000000 nM T16347 CSZB36 44329839 IC50 > 100000 nM T16347 CG7L1F 44329967 IC50 = 97000 nM T16347 C1PD9M 44332737 IC50 = 46000 nM T16347 CXF89O 44332885 IC50 = 19000 nM T16347 CV4I6P 44332900 IC50 = 18000 nM T16347 CI2U3R 44332905 IC50 = 20000 nM T16347 CHSE86 44332906 Ki = 17000 nM T16347 C8BU7F 44332907 IC50 = 25000 nM T16347 CNQU65 44332925 IC50 = 30000 nM T16347 CIM14F 44332928 IC50 = 24000 nM T16347 C1V7WS 44334321 Ki = 2800 nM T16347 C9PL7F 44334324 Ki = 220000 nM T16347 CEL2Q6 44334377 Ki = 9900 nM T16347 C8EPZ4 44334378 Ki = 760000 nM T16347 C39FED 44336385 Ki > 200000 nM T16347 CKE4U1 44336395 Ki = 2200 nM T16347 C92ZEG 44336558 Ki = 48600 nM T16347 CF0U7E 44336592 Ki = 2089.3 nM T16347 CF3R6Y 44336593 Ki = 1698.24 nM T16347 C8YMC6 44336749 Ki = 8400 nM T16347 CK84WX 44336750 Ki = 13800 nM T16347 CM17GK 44337392 IC50 = 85000 nM T16347 CXJO75 44337399 IC50 = 20000 nM T16347 CQV1I5 44337400 IC50 > 100000 nM T16347 CZQ8F0 44337401 IC50 = 10000 nM T16347 CZ79HK 44337402 IC50 > 100000 nM T16347 C75MSY 44337409 IC50 > 100000 nM T16347 CUD0O4 44337410 IC50 > 100000 nM T16347 C84VJN 44337423 IC50 = 51000 nM T16347 CQ3F5T 44337439 IC50 = 58000 nM T16347 CQN51Y 44337440 IC50 = 98000 nM T16347 C7X2CV 44337441 IC50 > 100000 nM T16347 C91ALN 44337454 IC50 > 100000 nM T16347 CTVW60 44337518 IC50 = 35000 nM T16347 CLW6G3 44337519 IC50 = 32000 nM T16347 C78WUC 44337562 IC50 > 100000 nM T16347 CRT7I6 44337574 IC50 = 58000 nM T16347 C5A9TD 44337575 IC50 > 100000 nM T16347 C7S3VN 44337581 IC50 = 58000 nM T16347 CC1K8N 44337589 IC50 > 100000 nM T16347 C6K3MN 44337596 IC50 = 83000 nM T16347 CG4X5N 44337597 IC50 = 90000 nM T16347 C6YJ9T 44337604 IC50 = 59000 nM T16347 CM6NJ2 44337607 IC50 > 100000 nM T16347 C90YQX 44337608 IC50 = 20000 nM T16347 C9VCW0 44337612 IC50 > 100000 nM T16347 C1OW4N 44337711 IC50 = 38000 nM T16347 CVW17B 44337712 IC50 = 45000 nM T16347 CD06ZI 44337719 IC50 = 77000 nM T16347 CXRJ74 44337726 IC50 > 100000 nM T16347 CNZ12Q 44337727 IC50 = 49000 nM T16347 C0I5NO 44337786 IC50 = 36000 nM T16347 CTRH27 44337799 IC50 > 100000 nM T16347 CV6U7P 44337816 IC50 > 100000 nM T16347 CN8GZ9 44340071 IC50 = 35000 nM T16347 C63UME 44340082 IC50 = 320000 nM T16347 C2J6MN 44340083 IC50 = 640000 nM T16347 CK0IF9 44340098 IC50 = 175000 nM T16347 CG8QA6 44340103 IC50 = 15000 nM T16347 C1T7UD 44340309 IC50 = 250000 nM T16347 C91NAV 44340331 IC50 = 435000 nM T16347 C5TF4H 44342137 IC50 = 41500 nM T16347 C4DW3U 44343960 IC50 = 15000 nM T16347 CFX1R5 44344024 Ki = 125892.54 nM T16347 CYX40O 44344614 IC50 = 130000 nM T16347 C6N7YQ 44345096 IC50 = 1410000 nM T16347 CLFE34 44345295 IC50 = 350000 nM T16347 CX28CS 44345402 IC50 = 1050000 nM T16347 C4M8ZC 44351283 Ki > 200000 nM T16347 C3GF2D 44351338 Ki > 200000 nM T16347 CJ5ZR3 44351395 Ki = 6100 nM T16347 CVTD37 44351411 Ki > 200000 nM T16347 CK1MU0 44351419 Ki > 200000 nM T16347 CO3RS9 44351420 Ki > 200000 nM T16347 CFLT90 44351505 Ki = 2000 nM T16347 C8C1IX 44358754 Ki = 12000 nM T16347 CGB0R8 44358930 Ki = 2200 nM T16347 CT20HY 44359237 Ki = 107151.93 nM T16347 C5YV1R 44359299 Ki = 37000 nM T16347 CS48HB 44360567 Ki = 930 nM T16347 CEG45Y 44361213 Ki = 1300000 nM T16347 CI82BW 44361260 Ki = 410000 nM T16347 CG4QM7 44361262 Ki = 1300000 nM T16347 C4LG7N 44361408 Ki = 1100000 nM T16347 CUG96K 44362351 IC50 = 83176377.11 nM T16347 CJM5P0 44362536 IC50 = 691830970.9 nM T16347 C6UXY7 44362554 IC50 = 46773514.13 nM T16347 CT17AE 44362616 IC50 = 707945784.4 nM T16347 C5ZWT7 44362646 IC50 = 70794578.44 nM T16347 C1KT0E 44362647 IC50 = 89125093.81 nM T16347 CTDB41 44362675 IC50 = 46773514.13 nM T16347 CE5A1P 44366440 IC50 = 135900 nM T16347 C5BEM3 44366445 IC50 = 778900 nM T16347 C5PGV2 44366478 IC50 = 128300 nM T16347 CXTA56 44366499 IC50 = 175700 nM T16347 CT35EW 44366675 IC50 = 449900 nM T16347 CH59XT 44366691 IC50 = 77500 nM T16347 CI0W6J 44366696 IC50 = 451400 nM T16347 C78OQD 44385071 Ki = 870 nM T16347 C3ZHV0 44385223 Ki = 700 nM T16347 C4KX3B 44386283 Ki = 1400 nM T16347 CN4WG2 44395083 Ki = 41000 nM T16347 CU4YM6 44395170 IC50 = 16000 nM T16347 CK4EI7 44396184 Ki = 18 nM T16347 CZGJ05 44397369 IC50 = 2800 nM T16347 C2ID8K 44397469 IC50 = 12000 nM T16347 CM0FQ8 44397470 IC50 = 24000 nM T16347 CK1NL8 44397522 IC50 > 100000 nM T16347 CC9HO5 44397523 IC50 > 100000 nM T16347 C7M6YB 44397524 IC50 > 100000 nM T16347 CPJ0D7 44397525 IC50 > 100000 nM T16347 C59QAC 44397526 IC50 = 4300 nM T16347 CI49PC 44397704 IC50 = 6400 nM T16347 C2R9MT 44397705 IC50 = 4300 nM T16347 CO16QX 44397838 IC50 = 4600 nM T16347 CS56NW 44397839 IC50 = 3100 nM T16347 CU26KL 44397840 IC50 = 3800 nM T16347 CEYQ42 44397841 IC50 = 13000 nM T16347 C50CFT 44397842 IC50 = 23000 nM T16347 CMQ9B1 44397962 IC50 = 2900 nM T16347 C53CWH 44398213 IC50 = 52480746.02 nM T16347 C1YE4I 44398266 IC50 = 52480746.02 nM T16347 CH8QB3 44398268 IC50 = 912010839.4 nM T16347 CT8PM0 44398363 IC50 = 776247116.6 nM T16347 CL4CY8 44398425 IC50 = 38018939.63 nM T16347 CS97BF 44399816 IC50 = 132000 nM T16347 CQ9F6M 44399819 IC50 = 203000 nM T16347 C34GDN 44399820 IC50 = 138000 nM T16347 CWU5E2 44404292 IC50 = 12000 nM T16347 C2TU6L 44404293 Ki = 98 nM T16347 CH7R0M 44404294 IC50 = 35 nM T16347 CWI10X 44404295 IC50 = 60 nM T16347 CWR1F2 44404296 IC50 = 1100 nM T16347 CRV1X5 44404297 Ki = 14 nM T16347 C0L1ZX 44404304 IC50 = 7000 nM T16347 CE72TH 44404305 Ki = 1100 nM T16347 CA0PF5 44404306 IC50 = 67500 nM T16347 CJ82YR 44404307 IC50 = 13700 nM T16347 CS1O3F 44404314 IC50 = 6900 nM T16347 CO1KJ6 44404315 IC50 = 2300 nM T16347 CS4M5O 44404320 IC50 = 3000 nM T16347 CWY93G 44404324 IC50 = 3000 nM T16347 CX8Q0K 44404329 IC50 = 4000 nM T16347 C59EVO 44404333 IC50 = 1000 nM T16347 C2T5JV 44404334 IC50 = 4000 nM T16347 C5BA0T 44404335 IC50 = 5000 nM T16347 CCFO74 44404340 IC50 = 4000 nM T16347 CO1Y4E 44404346 IC50 = 1900 nM T16347 CZF87M 44404350 IC50 = 2900 nM T16347 C4VC6U 44404353 IC50 = 1600 nM T16347 CTD1E3 44404358 IC50 = 770 nM T16347 CM7P6I 44404359 IC50 = 630 nM T16347 CT4MN3 44404360 IC50 = 1100 nM T16347 CKOL29 44404361 Ki = 590 nM T16347 CJF1D7 44404366 IC50 = 1000 nM T16347 C2LUQ7 44404367 IC50 = 180 nM T16347 CEIX02 44404368 Ki = 56 nM T16347 CO5J0G 44404369 IC50 = 220 nM T16347 CUC78J 44404373 IC50 = 9000 nM T16347 CO6TD8 44404376 IC50 = 6800 nM T16347 CKO5A0 44405932 IC50 > 100000 nM T16347 C4JZ1E 44405933 IC50 > 100000 nM T16347 CBX34H 44405951 IC50 > 100000 nM T16347 CAJ5T4 44405958 IC50 > 100000 nM T16347 CSLQ50 44405959 IC50 > 100000 nM T16347 C0Q5NW 44406035 IC50 = 80600 nM T16347 CX28MD 44406938 IC50 = 140 nM T16347 C1W0DB 44406944 IC50 = 7820 nM T16347 CW3TZ7 44406948 IC50 = 1640 nM T16347 CNOH38 44406981 IC50 = 7550 nM T16347 CKC39T 44406982 IC50 = 1960 nM T16347 C6ME8A 44407008 IC50 = 5480 nM T16347 CK6B5F 44407009 IC50 = 8190 nM T16347 C3R8JN 44407025 IC50 = 3400 nM T16347 CK3NA2 44407033 IC50 = 270 nM T16347 C4VO7S 44407055 IC50 = 2160 nM T16347 CQI09L 44407075 IC50 = 5630 nM T16347 CKP6O4 44408701 IC50 = 1600 nM T16347 CYW68I 44409605 IC50 = 7220 nM T16347 CGX23J 44409674 IC50 = 7190 nM T16347 CTM56S 44409675 IC50 = 7570 nM T16347 C6E4UN 44409680 IC50 = 4550 nM T16347 C25MUW 44409681 IC50 = 4110 nM T16347 CTL17C 44409833 IC50 = 7630 nM T16347 CB31QM 44409834 IC50 = 27160 nM T16347 CY6QB9 44409856 IC50 = 9050 nM T16347 C23ERY 44409919 IC50 = 19080 nM T16347 C56DNZ 44409999 IC50 = 10400 nM T16347 C70AZY 44410062 Ki = 72500 nM T16347 CF26CD 44410095 Ki = 27500 nM T16347 CJB6A7 44411589 IC50 > 30000 nM T16347 C4WI2K 44411623 IC50 > 30000 nM T16347 CE09UY 44411628 IC50 > 30000 nM T16347 CH64PJ 44411983 IC50 = 4900 nM T16347 C39UCN 44412819 IC50 = 340 nM T16347 C5P9FE 44412820 IC50 = 18 nM T16347 CY4D8H 44412833 IC50 = 15 nM T16347 CG6FM9 44412834 IC50 > 10000 nM T16347 CS45CR 44412846 IC50 = 110 nM T16347 CJCG57 44412858 IC50 = 240 nM T16347 CS07XV 44412859 IC50 = 140 nM T16347 CQHG97 44412872 IC50 = 280 nM T16347 CWC94K 44412885 IC50 = 160 nM T16347 CHQ92F 44412886 IC50 = 110 nM T16347 C6D8CL 44412891 IC50 = 76 nM T16347 C6MGY5 44412899 IC50 = 72 nM T16347 CONE93 44412900 IC50 = 190 nM T16347 C4I1DX 44412914 IC50 = 79 nM T16347 C6WDS5 44412919 IC50 = 16 nM T16347 CIF14B 44412937 IC50 = 51 nM T16347 CKL74J 44412939 IC50 = 18 nM T16347 CU91SR 44412974 IC50 = 10 nM T16347 CVX07M 44412998 IC50 = 32 nM T16347 CHG82C 44413042 IC50 = 120 nM T16347 CYQV74 44413043 IC50 = 53 nM T16347 COAG59 44413044 IC50 = 140 nM T16347 C09BXY 44413045 IC50 = 150 nM T16347 CEBD54 44413046 IC50 = 140 nM T16347 C8A4ZU 44413059 IC50 = 130 nM T16347 CA6K3X 44413060 IC50 = 460 nM T16347 CXM01H 44413062 IC50 = 50 nM T16347 COG2K8 44413994 Ki = 10000 nM T16347 CJUM36 44415112 IC50 > 100000 nM T16347 C2UD5Y 44419403 IC50 = 213800 nM T16347 C4SCY8 44422131 Ki = 37000 nM T16347 C2W3LF 44422132 Ki = 27500 nM T16347 CP67GJ 44422146 Ki = 45000 nM T16347 CA1LS2 44422179 Ki = 54000 nM T16347 CEFS05 44424282 IC50 = 380000 nM T16347 CL70RB 44424648 IC50 > 60000 nM T16347 CHDV14 44424650 IC50 = 18200 nM T16347 C8B7ZW 44430396 IC50 > 1000000 nM T16347 C0BW1D 44432363 IC50 = 17500 nM T16347 CC84UP 44432364 IC50 = 15700 nM T16347 CHZV64 44432618 IC50 = 260000 nM T16347 CC2W4Q 44432619 IC50 = 101000 nM T16347 CQ72RJ 44432621 IC50 = 137500 nM T16347 CPRT18 44432624 IC50 = 190000 nM T16347 CU97AL 44432625 IC50 = 168000 nM T16347 CXF14S 44434443 IC50 = 18000 nM T16347 C4Z6WR 44434444 IC50 = 2800 nM T16347 C0BE4L 44434445 IC50 = 1100 nM T16347 C4MEY2 44434446 IC50 = 5500 nM T16347 CHU6D0 44434447 IC50 = 6500 nM T16347 CM49EU 44434448 IC50 = 10200 nM T16347 C46WAB 44434669 IC50 > 1000000 nM T16347 CWE78X 44434670 IC50 > 1000000 nM T16347 CW59BQ 44434671 IC50 = 300000 nM T16347 CN7CE3 44434672 IC50 = 73000 nM T16347 CF9RC4 44434673 IC50 > 1000000 nM T16347 C9XA0L 44434674 IC50 = 93000 nM T16347 CFZ8I7 44434675 IC50 = 17000 nM T16347 CLU5N2 44434676 IC50 = 2200 nM T16347 CWN8V5 44434677 IC50 = 5000 nM T16347 CA9X5W 44434678 IC50 = 5700 nM T16347 CY4LH6 44434679 IC50 = 13000 nM T16347 CBUP13 44434680 IC50 = 5400 nM T16347 CH7PZ1 44434681 IC50 = 40000 nM T16347 C6OK9W 44439082 IC50 > 2500000 nM T16347 C7TWZ3 44439084 IC50 > 2500000 nM T16347 CV0X9U 44439085 IC50 > 2500000 nM T16347 C8JOI3 44439086 IC50 > 2500000 nM T16347 CKU5G6 44439087 IC50 > 2500000 nM T16347 CPX02D 44439088 IC50 > 2500000 nM T16347 C5TSG1 44439090 IC50 > 2500000 nM T16347 CG0V7P 44439092 IC50 > 2500000 nM T16347 C9JP2R 44439116 IC50 > 2500000 nM T16347 C4YFS0 44439117 IC50 > 2500000 nM T16347 CZ4UY9 44439118 IC50 = 210000 nM T16347 CE1W8K 44439119 IC50 > 2500000 nM T16347 CS3PR9 44439121 IC50 > 2500000 nM T16347 C6W4RJ 44439122 Ki = 210000 nM T16347 CJV46H 44439123 IC50 > 2500000 nM T16347 CR01JI 44439124 IC50 = 165000 nM T16347 CV76RK 44439125 IC50 > 2500000 nM T16347 CMFN16 44439126 IC50 > 2500000 nM T16347 CCH67J 44439127 IC50 > 2500000 nM T16347 C60JXG 44439128 IC50 > 2500000 nM T16347 CFZV35 44439129 Ki = 270000 nM T16347 CW0F8G 44439130 Ki = 20000 nM T16347 C5H3LS 44439131 Ki = 170000 nM T16347 C08BYZ 44439132 Ki = 120000 nM T16347 C5KU9I 44439133 Ki = 18000 nM T16347 CCB0P4 44439134 Ki = 1600 nM T16347 CY9JW5 44439135 Ki = 4600 nM T16347 C38CZJ 44439136 Ki = 1300 nM T16347 COVX74 44444618 IC50 = 1200 nM T16347 C4FD9Y 44444621 IC50 = 382000 nM T16347 CG7ZE3 44444622 IC50 = 176000 nM T16347 C73OHW 44444623 IC50 = 123000 nM T16347 C2ZQU4 44444624 IC50 = 59000 nM T16347 CL9N8K 44444625 IC50 = 32000 nM T16347 CKS7A8 44444627 IC50 = 27000 nM T16347 C1CQF2 44444633 IC50 = 37000 nM T16347 C8RLM0 44444636 IC50 = 105000 nM T16347 C40ITM 44444648 IC50 = 12000 nM T16347 CQ1M4W 44444651 IC50 = 23000 nM T16347 CLWO85 44444653 IC50 = 36000 nM T16347 CVYA12 44444655 IC50 = 10000 nM T16347 C7Q4FY 44444656 IC50 = 12000 nM T16347 CN9DJ4 44444657 IC50 = 500000 nM T16347 C96GTD 44446114 IC50 = 5030 nM T16347 CHX34E 44446115 IC50 = 240 nM T16347 CQD15S 44446116 IC50 = 700 nM T16347 CPGA64 44446117 IC50 = 540 nM T16347 CG3EB8 44446118 IC50 = 810 nM T16347 CCY8S6 44446119 IC50 = 930 nM T16347 CLF57A 44446120 IC50 = 660 nM T16347 CUR9P4 44446121 IC50 = 2900 nM T16347 CKI86T 44446122 IC50 = 150 nM T16347 C9OY2H 44446123 IC50 = 1300 nM T16347 C9BND2 44446124 IC50 = 210 nM T16347 CMUN01 44446125 IC50 = 64 nM T16347 C4AOP3 44446126 IC50 = 130 nM T16347 C6GUM2 44446127 IC50 = 800 nM T16347 CN4J7H 44446128 IC50 = 23 nM T16347 C9HBE4 44446129 IC50 = 160 nM T16347 CGC26X 44446130 IC50 = 110 nM T16347 CXJ18A 44446131 IC50 = 22 nM T16347 CAQ3Y8 44446132 IC50 = 100 nM T16347 C15BCG 44446133 IC50 = 300 nM T16347 CO2W7H 44446134 IC50 = 170 nM T16347 CCL8Y9 44446135 IC50 = 52 nM T16347 CXT8G1 44446136 IC50 = 200 nM T16347 CTK8B9 44446138 IC50 = 160 nM T16347 CBTD53 44446146 IC50 = 250 nM T16347 C9L0DV 44446159 IC50 = 180 nM T16347 C8D5BN 44446162 IC50 = 43 nM T16347 CJN0F3 44446164 IC50 = 260 nM T16347 CX51EZ 44446165 IC50 = 350 nM T16347 C9YX1C 44446168 IC50 = 120 nM T16347 C6I8BH 44446173 IC50 = 160 nM T16347 CUA4L1 44449556 IC50 = 510 nM T16347 CVD65P 44449557 IC50 = 1500 nM T16347 C74NTL 44449558 IC50 = 1300 nM T16347 C8OL7E 44449592 Ki = 179000 nM T16347 CJ1F2K 44449627 IC50 = 160 nM T16347 CV8DL7 44449628 IC50 = 7 nM T16347 CVZ04W 44449658 IC50 > 50000 nM T16347 CRJA86 44449698 IC50 = 16 nM T16347 CTSC68 44450221 IC50 = 63600 nM T16347 CY05UW 44450233 IC50 = 29100 nM T16347 CS43YR 44450234 IC50 = 232000 nM T16347 CY5L3C 44450244 IC50 > 250000 nM T16347 CMET71 44450245 IC50 = 173000 nM T16347 C5OC8H 44450247 IC50 > 250000 nM T16347 C15GLF 44450251 IC50 = 114000 nM T16347 CA7CB6 44450252 IC50 = 115000 nM T16347 C63FDU 44450253 IC50 = 12200 nM T16347 CCP2H6 44450263 IC50 = 80700 nM T16347 CA5BX2 44450264 IC50 = 4400 nM T16347 C6FC2U 44450265 IC50 = 76200 nM T16347 CK09NL 44450272 IC50 = 7900 nM T16347 CU01BF 44450273 IC50 = 4100 nM T16347 CZ5JI3 44450274 IC50 = 53800 nM T16347 CFIG07 44450283 IC50 = 57700 nM T16347 CHK7M2 44450284 IC50 = 38000 nM T16347 CAZ75L 44450285 IC50 = 137000 nM T16347 CY1X0B 44450287 IC50 = 19900 nM T16347 CR7B1T 44450291 IC50 > 250000 nM T16347 CA5LV0 44450292 IC50 = 198000 nM T16347 CB0FH6 44450294 IC50 = 230000 nM T16347 CPHE21 44450295 IC50 = 97100 nM T16347 CZE2X6 44450308 IC50 = 153000 nM T16347 C35PVL 44450309 IC50 = 29100 nM T16347 C6SUA3 44450310 IC50 = 74200 nM T16347 C8T9EW 44450317 IC50 = 237000 nM T16347 C4Q0WK 44450318 IC50 = 52100 nM T16347 C8RJ6W 44450319 IC50 > 250000 nM T16347 CRVU24 44450321 IC50 = 54100 nM T16347 CNLB76 44450331 IC50 = 77900 nM T16347 CJ7UM2 44450333 IC50 = 123000 nM T16347 CKA9T6 44450335 IC50 = 59600 nM T16347 C2FZ1E 44450343 IC50 = 60300 nM T16347 CZSX79 44450344 IC50 = 96800 nM T16347 C16PNM 44450352 IC50 = 51800 nM T16347 C0D4YU 44450353 IC50 = 27600 nM T16347 CNX63F 44450354 IC50 = 17700 nM T16347 C7GR3D 44450362 IC50 = 235000 nM T16347 C5ZU1W 44450363 IC50 = 13800 nM T16347 C7BPV1 44450364 IC50 > 250000 nM T16347 CDT5X4 44450373 IC50 = 10100 nM T16347 C2CT8R 44456685 Ki = 4500 nM T16347 C5J2HZ 44520379 IC50 = 5500 nM T16347 CPK2B3 44537949 IC50 = 2900 nM T16347 CWXT19 44537950 IC50 = 1500 nM T16347 CG16HZ 44537957 IC50 = 8800 nM T16347 CER40Q 44537958 IC50 = 4200 nM T16347 C9LIF8 44560647 IC50 = 6 nM T16347 C64RCZ 44560687 Ki = 10600 nM T16347 C2BWH1 44560689 Ki = 10300 nM T16347 C76BKL 44560691 Ki = 24 nM T16347 CJVL45 44560693 Ki = 3300 nM T16347 C4NGR1 44560695 Ki = 24 nM T16347 C76POH 44560697 IC50 = 10000 nM T16347 C3VQF5 44560744 IC50 = 44000 nM T16347 CKL18I 44562663 IC50 = 20430 nM T16347 CYCE47 44562664 IC50 = 27610 nM T16347 CAW16R 44562712 IC50 = 15950 nM T16347 C26ZAB 44562713 IC50 = 16550 nM T16347 C51QGN 44562714 IC50 = 1120 nM T16347 C7XP8B 44562715 IC50 = 2440 nM T16347 C3F8MD 44562716 IC50 = 2360 nM T16347 C49JDA 44562718 IC50 = 4130 nM T16347 C4VM5Z 44562925 IC50 = 4520 nM T16347 C1ATZ5 44562926 IC50 = 5270 nM T16347 C3R2HL 44563278 IC50 = 3310 nM T16347 CGI61Y 44563279 IC50 = 15440 nM T16347 C7GW0X 44563280 IC50 = 16350 nM T16347 CL15CQ 44563281 IC50 = 3090 nM T16347 C8GH6J 44563282 IC50 = 4760 nM T16347 CM18HZ 44563318 IC50 = 9200 nM T16347 CNT53M 44563343 IC50 = 8100 nM T16347 CR50UK 44563344 IC50 = 2100 nM T16347 C9PC6L 44563345 IC50 = 1330 nM T16347 CXR50S 44563346 IC50 = 880 nM T16347 CMF92J 44563347 IC50 = 780 nM T16347 CCE23Q 44563348 IC50 = 720 nM T16347 CGNY85 44563349 IC50 = 590 nM T16347 C3HDB9 44563372 IC50 = 570 nM T16347 C0ZE7Q 44563373 IC50 = 740 nM T16347 CRN37D 44563374 IC50 = 4620 nM T16347 C6RWF4 44563375 IC50 = 590 nM T16347 C4FC7K 44563376 IC50 = 550 nM T16347 CN89UB 44563377 IC50 = 560 nM T16347 COW78E 44563378 IC50 = 510 nM T16347 CXG7B2 44563379 IC50 = 610 nM T16347 CIRW95 44563380 IC50 = 570 nM T16347 C9R2OG 44563381 IC50 = 450 nM T16347 C4CX3J 44563382 IC50 = 550 nM T16347 CI6SG7 44563383 IC50 = 650 nM T16347 CQ97PD 44563384 IC50 = 530 nM T16347 CU4QC1 44563385 IC50 = 520 nM T16347 C0FN6C 44563386 IC50 = 600 nM T16347 CT94FG 44563387 IC50 = 440 nM T16347 C5Y7IK 44563388 IC50 = 660 nM T16347 CK9JV2 44563389 IC50 = 820 nM T16347 CM15VN 44563390 IC50 = 630 nM T16347 C73HRF 44563443 IC50 = 2890 nM T16347 CT2IV9 44563444 IC50 = 2670 nM T16347 C60MCT 44563445 IC50 = 2720 nM T16347 C35SXC 44563446 IC50 = 620 nM T16347 CDP45M 44563447 IC50 = 540 nM T16347 C8MXT3 44563448 IC50 = 150 nM T16347 CB6YK7 44563449 IC50 = 2850 nM T16347 CR46UO 44563511 IC50 = 71 ug.mL-1 T16347 C7MP5Y 44563570 IC50 = 530 nM T16347 C5Q2FM 44563588 IC50 = 34000 nM T16347 C7D5GS 44563589 IC50 = 30000 nM T16347 CBV8J9 44563590 IC50 = 13000 nM T16347 CP2H1Y 44563591 IC50 = 32000 nM T16347 C0Q8OC 44563592 IC50 = 64000 nM T16347 C5Q3WP 44563617 IC50 = 194000 nM T16347 C5I4ZO 44563618 IC50 = 125000 nM T16347 CHNU48 44563656 IC50 = 6000 nM T16347 C3LMP9 44563657 IC50 = 4000 nM T16347 C02YOA 44567037 IC50 = 17000 nM T16347 C31PNJ 44568935 IC50 > 30000 nM T16347 C6R5AB 44572192 IC50 = 2000 nM T16347 C8DX3F 44572209 IC50 = 1080 nM T16347 CYP60M 44572709 Ki = 29100 nM T16347 C8H7AW 44572965 IC50 = 17000 nM T16347 CKA6O7 44572966 IC50 = 6200 nM T16347 CM91XV 44573085 IC50 = 5000 nM T16347 C86QNW 44573086 IC50 = 900 nM T16347 CTNO02 44577536 IC50 = 1.9 ug.mL-1 T16347 C5BF2O 44577537 IC50 = 8.8 ug.mL-1 T16347 C2DBZ3 44578543 IC50 = 2000 nM T16347 C27TIC 44582365 IC50 = 1900 nM T16347 CNJ13R 44582366 IC50 = 1100 nM T16347 CW4Y0E 44582367 IC50 = 3800 nM T16347 CW74DT 44582392 IC50 = 1100 nM T16347 C2JBW6 44582393 IC50 = 14000 nM T16347 CKL5M7 44582394 IC50 = 1900 nM T16347 CH1YX2 44582395 IC50 = 35400 nM T16347 C48QVJ 44582421 IC50 = 30100 nM T16347 CI8XC7 44582422 IC50 = 32100 nM T16347 C8A5RD 44582423 IC50 = 33700 nM T16347 CDT8B9 44582424 IC50 = 19500 nM T16347 C9EJQ8 44588360 IC50 = 870 nM T16347 C0YA9X 44588361 IC50 = 880 nM T16347 CK8N5I 44588362 IC50 = 620 nM T16347 CGT50K 44588363 IC50 = 720 nM T16347 C16IXC 44589106 IC50 = 13900 nM T16347 CEBS52 44589107 IC50 > 60000 nM T16347 CC5Y3K 44589108 IC50 > 60000 nM T16347 CL59FI 44589132 IC50 = 14900 nM T16347 CMH4O3 44589217 IC50 > 60000 nM T16347 CZO2P9 44589218 IC50 = 19000 nM T16347 C68AOE 44589219 IC50 = 18200 nM T16347 CQ9P7O 44589231 IC50 > 60000 nM T16347 C0AKG5 44589232 IC50 > 60000 nM T16347 C5FKA0 44589233 IC50 > 60000 nM T16347 C8DU3P 44591657 IC50 = 72000 nM T16347 C2Z7QF 45266940 Ki = 630.96 nM T16347 C7W4QO 45266969 Ki = 10000 nM T16347 CT9LP2 45266987 Ki = 7943.28 nM T16347 CX53WK 45267150 IC50 = 3020 nM T16347 CSY91T 45267799 Ki = 3981.07 nM T16347 C4LE7A 45267803 Ki = 100000 nM T16347 C17VZQ 45267805 Ki = 25118.86 nM T16347 CNPV10 45267806 Ki = 251188.64 nM T16347 CVS7Z6 45267846 Ki = 251188.64 nM T16347 CQUX74 45267905 Ki = 3981.07 nM T16347 C6R5NH 45267906 Ki = 3162277.66 nM T16347 CHD5T6 45267908 IC50 = 22 nM T16347 CJR20X 45268689 Ki = 251.19 nM T16347 CU35MY 45268692 Ki = 251.19 nM T16347 CR31KA 45268722 Ki = 1995.26 nM T16347 CR8DU9 45268723 Ki = 7943.28 nM T16347 COE14I 45268794 Ki = 125892.54 nM T16347 C9TWX8 45268796 Ki = 50118.72 nM T16347 CD5F4R 45269556 Ki = 630957.34 nM T16347 CVF13L 45269583 Ki = 125892.54 nM T16347 C5B9IX 45269639 Ki = 1584.89 nM T16347 CO80VZ 45270371 Ki = 10000 nM T16347 C7ESN5 45270378 Ki = 199526.23 nM T16347 CGE76Y 45270379 Ki = 630.96 nM T16347 C5YUN4 45270385 Ki = 7943.28 nM T16347 C4J8KF 45270471 Ki = 316227.77 nM T16347 C8S5KT 45270472 Ki = 39810.72 nM T16347 CM60XP 45270473 Ki = 6309.57 nM T16347 C6JS2G 45270474 Ki = 5011.87 nM T16347 CDC8Z2 45271196 Ki = 7943.28 nM T16347 C5AY1W 45271201 Ki = 3981.07 nM T16347 CE53OG 45271202 Ki = 158489.32 nM T16347 CIC47Z 45271203 Ki = 3981.07 nM T16347 C2CRX1 45271207 Ki = 398.11 nM T16347 CQLI76 45271212 Ki = 19952.62 nM T16347 C6SPA3 45271248 Ki = 630.96 nM T16347 C1HR5E 45271304 Ki = 1258.93 nM T16347 CD9EX1 45271305 Ki = 19952.62 nM T16347 C9EUS6 45271564 IC50 = 610 nM T16347 CD6Y9T 45271762 IC50 = 41000 nM T16347 CUW28D 45272102 Ki = 1000000 nM T16347 C59GPO 45272108 Ki = 12589.25 nM T16347 CU8P2G 45272110 Ki = 1995.26 nM T16347 CR5JQ3 45272190 Ki = 501187.23 nM T16347 C67JKG 45272934 Ki = 3981.07 nM T16347 CLR98Q 45272946 Ki = 12589.25 nM T16347 CJ3C9Q 45273035 IC50 = 1700 nM T16347 CXTO38 45273054 Ki = 6309.57 nM T16347 CL1U8M 45273157 IC50 = 7420 nM T16347 C29SCR 45273528 IC50 = 28000 nM T16347 C09UXA 45375877 IC50 > 30000 nM T16347 C41ADU 45469287 IC50 = 9700 nM T16347 C3TKO9 45474108 IC50 = 8900 nM T16347 C9IN0G 45482806 IC50 = 8000 nM T16347 C45ARN 45482812 IC50 = 14000 nM T16347 CUYZ60 45482821 IC50 = 8000 nM T16347 CU9W2R 45482822 IC50 = 8000 nM T16347 CO1GI5 45482833 Ki = 2100 nM T16347 C6CH8J 45482834 IC50 = 15000 nM T16347 C1R2AV 45482835 IC50 = 5000 nM T16347 C46GSV 45482841 IC50 = 15000 nM T16347 CBI86P 45482842 IC50 = 9000 nM T16347 CG93SP 45482853 IC50 = 8000 nM T16347 CEY70L 45482857 IC50 = 6000 nM T16347 CYRC54 45482878 IC50 = 1920 nM T16347 C08CXZ 45482880 IC50 = 5440 nM T16347 CBO7R6 45482882 IC50 = 1780 nM T16347 CK98JB 45482885 IC50 = 2600 nM T16347 CQ5U3C 45482886 IC50 = 1390 nM T16347 C8Z7HX 45482894 IC50 = 2730 nM T16347 CCKE09 45482895 IC50 = 1650 nM T16347 CS28XV 45482896 IC50 = 1480 nM T16347 CWPI45 45482897 IC50 = 1750 nM T16347 CJT89W 45482898 IC50 = 640 nM T16347 CDRY08 45482899 IC50 = 810 nM T16347 CP68TN 45482901 IC50 = 2610 nM T16347 C45RQB 45485201 IC50 = 2700 nM T16347 CD3FM1 45487322 IC50 = 19200 nM T16347 CB7K3Z 45487346 IC50 = 17300 nM T16347 C15VOK 45487351 IC50 = 19400 nM T16347 C57BKJ 45487352 IC50 = 29200 nM T16347 C45AFN 46186815 Ki > 100000 nM T16347 C0DX6B 46209991 IC50 = 20700 nM T16347 C7YZA3 46228445 IC50 = 3000 nM T16347 CBJ7Z6 46228829 IC50 = 6700 nM T16347 CI3LQ4 46228831 IC50 = 5400 nM T16347 CCX49G 46228871 IC50 = 6800 nM T16347 CYD0N5 46228872 IC50 = 8500 nM T16347 CK0VT9 46228873 IC50 = 4800 nM T16347 C1JPB2 46228874 IC50 = 4600 nM T16347 CR1H8C 46228919 IC50 = 5000 nM T16347 CE1M2T 46228921 IC50 = 2100 nM T16347 CWN2P8 46228922 IC50 = 8700 nM T16347 CM0P8E 46229954 IC50 > 20000 nM T16347 C6CO2K 46229997 IC50 = 5 nM T16347 CL8UH0 46230053 IC50 = 3200 nM T16347 C6M2WF 46230054 IC50 = 16 nM T16347 C97XCE 46230105 IC50 = 32 nM T16347 CYF1D6 46230106 IC50 = 27 nM T16347 CJ3ZC9 46230107 IC50 = 23 nM T16347 CG0LP4 46230108 Ki = 4300 nM T16347 C6DQT4 46230153 IC50 = 14 nM T16347 CM97RA 46230154 IC50 = 12.6 nM T16347 CNE8V2 46230155 IC50 = 130 nM T16347 CX2T7S 46230200 IC50 = 8000 nM T16347 C28XVK 46231918 IC50 > 24000 nM T16347 C17TNY 46499243 IC50 = 15000 nM T16347 CHZ1N5 46703740 IC50 > 23000 nM T16347 CLGB06 46830252 IC50 > 10000000 nM T16347 C81CPM 46861833 IC50 = 350 nM T16347 C0A9LD 46861834 IC50 = 410 nM T16347 CT1S2F 46879574 IC50 = 40500 nM T16347 C8R5KT 46879575 IC50 = 65500 nM T16347 CC2N5R 46879576 IC50 = 70600 nM T16347 C3B5CI 46879577 IC50 = 76200 nM T16347 CBRL16 46879997 IC50 > 30000 nM T16347 C1SJG2 46882139 IC50 = 52400 nM T16347 CBX1Y7 46882140 IC50 = 62100 nM T16347 CEB2A7 46882183 IC50 = 56700 nM T16347 C9KF2J 46882184 IC50 = 24500 nM T16347 C3KN8B 46882185 IC50 = 36200 nM T16347 CA8T4N 46882186 IC50 = 82700 nM T16347 CEV34O 46882187 IC50 = 90400 nM T16347 C83GCS 46882340 Ki = 100 nM T16347 CAYL45 46882341 IC50 = 17000 nM T16347 CHQC68 46882382 IC50 = 590 nM T16347 C0OHS1 46887676 IC50 = 7160 nM T16347 CPEG29 46888174 IC50 = 1560 nM T16347 COD47H 46888363 IC50 = 7490 nM T16347 CK5IM2 46890075 IC50 = 120.23 nM T16347 CHA51I 46890630 IC50 = 2187.76 nM T16347 CK1GZ9 46906768 IC50 = 5300 nM T16347 CSO81B 46906769 IC50 = 12690 nM T16347 CWD54F 46906770 IC50 = 4600 nM T16347 CI0VC8 46906771 IC50 = 4140 nM T16347 C5SF3W 46906772 IC50 = 2750 nM T16347 C8Z1HV 46906773 IC50 = 2360 nM T16347 C7BZ1E 46906774 IC50 = 1900 nM T16347 C1HF7I 46906775 IC50 = 2080 nM T16347 C2PSM6 46906776 IC50 = 2610 nM T16347 C2HVZ6 46906777 IC50 = 1960 nM T16347 CSW3O5 46906778 IC50 = 1700 nM T16347 CBS74A 46906779 IC50 = 1420 nM T16347 CHC1W4 46906780 IC50 = 1620 nM T16347 C95DQW 46906781 IC50 = 330 nM T16347 CC82OY 46906782 IC50 = 270 nM T16347 CNEC74 46906783 IC50 = 500 nM T16347 CB3VQ1 46906784 IC50 = 13120 nM T16347 C4DM9B 46906786 IC50 = 11590 nM T16347 C8W6GX 46906787 IC50 = 6580 nM T16347 CFY21C 46906838 IC50 = 11300 nM T16347 C6RFL0 46910728 IC50 = 2900 nM T16347 C4M5OR 46913133 IC50 = 480 nM T16347 CE4J2Q 46933001 IC50 = 201 nM T16347 C2Z1XN 46933002 IC50 = 185 nM T16347 CGW4J9 46933003 IC50 = 257 nM T16347 CH9K7C 46933145 IC50 = 82 nM T16347 C0VH2C 46933146 IC50 = 121 nM T16347 C9VM5F 46933147 IC50 = 280 nM T16347 C4Z0CS 46933148 IC50 = 187 nM T16347 C6BIA2 46933149 IC50 = 388 nM T16347 CH92OW 46933294 IC50 = 395 nM T16347 CQ0FX3 46933295 IC50 = 425 nM T16347 CX8VZ6 46933442 IC50 = 620 nM T16347 CZIO39 46933443 IC50 = 551 nM T16347 CDR12P 46934435 IC50 = 25500 nM T16347 CWN9O2 46938438 IC50 = 220 nM T16347 CG1WI4 46938543 IC50 = 1600 nM T16347 CC65EH 46938544 IC50 = 490 nM T16347 C8K5PM 46938545 IC50 = 1200 nM T16347 C5P0NH 49796540 Ki = 8000000 nM T16347 C3A2BY 49796575 Ki = 16000 nM T16347 CGYM23 49796578 IC50 = 118000 nM T16347 CMA49Q 49796582 IC50 = 29000 nM T16347 C2IU1Z 49796692 IC50 = 3900 nM T16347 CT95HV 49797129 IC50 = 37000 nM T16347 C3M0WE 49797130 IC50 = 36700 nM T16347 C6E1OB 49797131 IC50 = 285700 nM T16347 C6NFP9 49797132 IC50 = 271200 nM T16347 CW3R6H 49797133 IC50 = 83600 nM T16347 C9L1NR 49797134 IC50 = 164000 nM T16347 CSWL06 49797135 IC50 = 153500 nM T16347 CNO54R 49797136 IC50 = 24900 nM T16347 C8EI0A 49797137 IC50 > 500000 nM T16347 CFN39K 49797138 IC50 = 148000 nM T16347 CR7H1S 49797139 IC50 = 134800 nM T16347 C2S9QH 49797140 IC50 = 95300 nM T16347 C73SHZ 49797141 IC50 = 64400 nM T16347 C7YPR2 49797154 IC50 = 16200 nM T16347 CZR0Y3 49797156 IC50 = 2300 nM T16347 C4V3AU 49797169 IC50 = 12800 nM T16347 CSBV96 50898774 IC50 = 1300 nM T16347 CV53DN 50908842 IC50 = 2.97 ug.mL-1 T16347 CF4D0K 50908843 IC50 = 2.66 ug.mL-1 T16347 C4AEZ1 50925509 IC50 = 205 nM T16347 C95QWO 50925510 IC50 = 190 nM T16347 CK1YX2 50941649 IC50 = 11500 nM T16347 C1PJL0 50941745 IC50 = 214 nM T16347 CRF1O3 50942131 IC50 = 217 nM T16347 C2NJ3B 51003508 IC50 = 14000 nM T16347 C6UHD8 51042112 Ki = 5100 nM T16347 CA8PE3 52325746 IC50 = 13800 nM T16347 CV3L9R 52940547 Ki = 1.4 nM T16347 CN4B2Q 52940585 IC50 = 177 nM T16347 C7M5ZG 52940863 IC50 = 515 nM T16347 C2VK4D 52943422 IC50 = 102 ug.mL-1 T16347 CQ19GI 52943423 IC50 = 65.3 ug.mL-1 T16347 CE1BA6 52945264 IC50 = 1500 nM T16347 C3QN8K 52947089 IC50 = 69.8 ug.mL-1 T16347 C5W4BT 52949107 IC50 = 3200 nM T16347 CUN0L6 52952499 IC50 = 2230 nM T16347 C7DO2K 53248945 IC50 = 17200 nM T16347 CZF5T9 53262772 IC50 = 23810 nM T16347 CTY08P 53262773 IC50 = 39670 nM T16347 CMYL23 53307612 IC50 = 2450 nM T16347 CMDB84 53316640 IC50 = 31200 nM T16347 C9GVU5 53317937 IC50 = 28100 nM T16347 CV4QD5 53317938 IC50 = 5100 nM T16347 C3QSB2 53318103 IC50 = 6390 nM T16347 CWT10N 53319270 IC50 > 50000 nM T16347 CRC82E 53320578 IC50 = 42300 nM T16347 C8Y4KW 53320579 IC50 = 8300 nM T16347 CF35GK 53320580 IC50 = 7000 nM T16347 C04CYS 53320581 IC50 > 50000 nM T16347 CJF79D 53321379 IC50 = 21860 nM T16347 CBI29Z 53321875 IC50 = 11200 nM T16347 CWN60J 53322036 IC50 = 3120 nM T16347 C3COY2 53322976 IC50 = 4110 nM T16347 C94WKB 53324565 IC50 = 16800 nM T16347 CZ6M2C 53324714 IC50 = 4610 nM T16347 CZD9L1 53324788 IC50 = 63900 nM T16347 C1EM5Y 53340938 IC50 = 2020 nM T16347 CF1RY7 53354232 IC50 = 1500 nM T16347 CE84SX 53355017 IC50 = 6600 nM T16347 C68LGK 53357588 IC50 = 41000 nM T16347 C68RVC 53357980 IC50 = 16360 nM T16347 CXDE41 53357981 IC50 = 14930 nM T16347 C1BOR3 53357982 IC50 = 13920 nM T16347 CL0HI5 53361713 IC50 = 5 nM T16347 C25RBT 53371735 IC50 = 2000 nM T16347 C2X9PM 53371736 IC50 = 630 nM T16347 CUQ25O 53371738 IC50 = 1500 nM T16347 CCNG89 54576098 IC50 = 2490 nM T16347 CV3YH5 54576318 IC50 = 2790 nM T16347 C4CAU1 54576319 IC50 = 1250 nM T16347 CYK80P 54576320 IC50 = 2590 nM T16347 CKD3W9 54576321 IC50 = 1770 nM T16347 C1P4QM 54576322 IC50 = 1570 nM T16347 C5LVA7 54580436 IC50 = 24160 nM T16347 C5D8AH 54580437 IC50 = 2500 nM T16347 CYBX30 54580826 IC50 > 30000 nM T16347 COYB06 54580827 IC50 = 2600 nM T16347 CVA15G 54580828 IC50 = 8000 nM T16347 CH82AU 54580829 IC50 = 4400 nM T16347 CORT50 54580846 IC50 = 1900 nM T16347 CN15QH 54580847 IC50 = 7000 nM T16347 CO3H2F 54581227 Ki = 26 nM T16347 C4IM5J 54581228 IC50 = 220 nM T16347 CNY9Q2 54581869 IC50 = 3500 nM T16347 CWD95V 54581870 IC50 = 2300 nM T16347 C4TK5F 54581871 IC50 = 18400 nM T16347 C28IEY 54581872 IC50 = 3400 nM T16347 C7BL4P 54581873 IC50 = 4500 nM T16347 CB3J6Q 54581874 IC50 = 4900 nM T16347 CH3A9I 54581875 IC50 = 3400 nM T16347 CMJ23F 54581906 IC50 = 2900 nM T16347 CZTS41 54582253 IC50 = 20 nM T16347 CV6HX5 54582254 IC50 = 40 nM T16347 CW1J5C 54582454 IC50 = 4400 nM T16347 CXO40T 54582455 IC50 = 5250 nM T16347 CWA9N5 54582456 IC50 = 31110 nM T16347 C7AGY5 54582457 IC50 = 4300 nM T16347 CATW95 54582802 IC50 = 13700 nM T16347 CYT41C 54582803 IC50 = 30000 nM T16347 CGF69R 54582804 IC50 = 11300 nM T16347 CNAD42 54583803 IC50 = 11100 nM T16347 CQ19TI 54583804 IC50 = 6200 nM T16347 CK5VL7 54583805 IC50 = 6800 nM T16347 CHFM90 54583806 IC50 = 6000 nM T16347 C80OEJ 54583841 IC50 = 2900 nM T16347 C2M9TC 54584394 IC50 = 5440 nM T16347 C5LJP0 54584395 IC50 = 25280 nM T16347 CT4H1S 54584396 IC50 = 37310 nM T16347 CSY6A0 54584397 IC50 = 9100 nM T16347 CY9RI3 54584776 IC50 = 9900 nM T16347 CD3Z8Y 54584777 IC50 = 4900 nM T16347 CP1GY0 54584778 IC50 = 2400 nM T16347 C2FA9U 54584779 IC50 = 13900 nM T16347 CJC09X 54584801 IC50 = 10300 nM T16347 C78KIM 54585348 IC50 = 22360 nM T16347 C3TGI2 54585350 IC50 = 56890 nM T16347 CTY1K4 54585717 IC50 = 4200 nM T16347 CRP58G 54585718 IC50 > 30000 nM T16347 C6WU1G 54585719 IC50 = 26400 nM T16347 CK32UJ 54585720 IC50 = 6800 nM T16347 C8TXF1 54585744 IC50 = 2600 nM T16347 CH1XC7 54586309 IC50 = 3310 nM T16347 CU69PW 54586696 IC50 = 10800 nM T16347 C4W1MC 54586697 IC50 = 2700 nM T16347 CK2QD9 54586698 IC50 = 6300 nM T16347 C6S2NQ 54587338 IC50 = 28030 nM T16347 C0FL4Q 54587339 IC50 = 3460 nM T16347 CA16KR 54587340 IC50 = 26710 nM T16347 CEY59T 54587733 IC50 = 2900 nM T16347 CE8PL0 54587734 IC50 = 15200 nM T16347 CBWY45 54587735 IC50 = 3500 nM T16347 CO31SZ 54587736 IC50 = 7100 nM T16347 C35SHL 54587737 IC50 = 6900 nM T16347 C7Q1PF 54587761 IC50 = 5300 nM T16347 C93LZF 54682873 IC50 = 1500 nM T16347 CQ30US 54685915 IC50 = 700 nM T16347 CS9NC4 54693142 IC50 > 100000 nM T16347 CZ82GO 54695794 IC50 = 28700 nM T16347 C87DUR 54695884 IC50 = 14600 nM T16347 CT7S1R 54697955 IC50 = 1000 nM T16347 CW3M8N 54706178 IC50 = 72700 nM T16347 C73TSH 54718593 IC50 = 400 nM T16347 CZ83RW 54751676 IC50 > 100000 nM T16347 CON5G1 54751677 IC50 = 25000 nM T16347 C9MP3W 54751678 IC50 > 100000 nM T16347 CCK72T 54751679 IC50 > 100000 nM T16347 C7K4GA 54757715 IC50 > 120000 nM T16347 C0NM6I 54757716 IC50 > 120000 nM T16347 CPX4I2 54757717 IC50 > 120000 nM T16347 C5OK3S 54757809 IC50 > 120000 nM T16347 C0DO1G 54757810 IC50 > 120000 nM T16347 CK49WP 54757811 IC50 = 100000 nM T16347 C5AQ8R 54757812 IC50 > 120000 nM T16347 CSPR73 54757813 IC50 > 120000 nM T16347 CK6Z3T 54757904 IC50 = 73000 nM T16347 C96NIW 54757905 IC50 > 100000 nM T16347 CT43AJ 54757906 IC50 > 100000 nM T16347 C93VEA 54758002 IC50 = 48000 nM T16347 C86LHU 54758003 IC50 > 100000 nM T16347 C79UJG 54758004 IC50 > 100000 nM T16347 C30WXK 54758005 IC50 > 100000 nM T16347 CB1QG9 54768265 IC50 > 300000 nM T16347 C6HW3Z 54768267 IC50 = 11070 nM T16347 CFSR86 54768269 IC50 = 24730 nM T16347 CB96GH 54768270 IC50 = 6550 nM T16347 CJH2Q3 54768305 IC50 = 14280 nM T16347 CF2J3U 54768306 IC50 = 21690 nM T16347 C1GDN4 54768308 IC50 = 7910 nM T16347 CM8H3X 54768309 IC50 = 10800 nM T16347 CB80UX 54768349 IC50 = 11390 nM T16347 C2R5JW 54768350 IC50 = 8880 nM T16347 C1VCJ9 54768351 IC50 = 3380 nM T16347 CF7X2K 54768352 IC50 = 4000 nM T16347 C48KOI 54768353 IC50 = 4220 nM T16347 CK3W0Z 54768391 IC50 = 4710 nM T16347 C01LRT 54768392 IC50 = 8150 nM T16347 C8DLG4 54768393 IC50 = 5900 nM T16347 CPGC13 54768394 IC50 = 4450 nM T16347 CVA04X 54768395 IC50 = 6480 nM T16347 CNZY43 56589511 IC50 > 10000000 nM T16347 C53XYO 56589513 IC50 > 10000000 nM T16347 CMY6E8 56598867 IC50 = 7800 nM T16347 CX6BM4 56600675 IC50 = 5900 nM T16347 C1NZJ0 56655196 IC50 = 2490 nM T16347 C0NGL1 56655720 IC50 = 8630 nM T16347 CS1ED4 56655721 IC50 = 2810 nM T16347 CUTW43 56655722 IC50 = 4260 nM T16347 CEC0N8 56659163 IC50 > 100000 nM T16347 CJG32W 56659993 Ki = 2100 nM T16347 CHM5V3 56660070 IC50 = 67800 nM T16347 CUF4X8 56662949 IC50 = 9000 nM T16347 C9NQ3F 56666422 IC50 = 19000 nM T16347 CF7P6Y 56666423 IC50 = 11000 nM T16347 C1U4BY 56668316 IC50 = 16600 nM T16347 CGW9Z5 56668381 IC50 = 245000 nM T16347 CWE5R8 56669528 IC50 = 15200 nM T16347 CX24DV 56669529 IC50 = 98100 nM T16347 C7V5YN 56669840 IC50 = 10000 nM T16347 C7J4QM 56669841 IC50 = 1400 nM T16347 C6WB8H 56669842 IC50 = 12000 nM T16347 C1Z4LT 56669843 IC50 = 2000 nM T16347 CHOF39 56670422 IC50 = 18500 nM T16347 CI9R8M 56670423 IC50 > 120000 nM T16347 C0N2KF 56671798 IC50 = 64600 nM T16347 CLN96K 56671799 IC50 = 19700 nM T16347 CNB8X7 56673037 IC50 = 35800 nM T16347 CSZ61X 56673038 IC50 > 100000 nM T16347 CWZ63T 56673321 IC50 = 4000 nM T16347 CKE05S 56673322 IC50 = 12000 nM T16347 CL3N0K 56673907 IC50 = 22300 nM T16347 CAL96I 56673908 IC50 = 7100 nM T16347 C90ARL 56675207 IC50 = 38700 nM T16347 CH4EO3 56675208 IC50 = 28900 nM T16347 CWXK83 56675796 IC50 > 300000 nM T16347 C9ZCA7 56676666 IC50 = 16000 nM T16347 CCH18Y 56676667 IC50 = 4000 nM T16347 CDJ4E5 56678312 Ki = 11000 nM T16347 CNL57P 56678510 IC50 = 19300 nM T16347 C1HS2O 56679982 IC50 = 9000 nM T16347 C2ZGS5 56679983 IC50 = 8000 nM T16347 CB8G5A 56679984 IC50 = 136000 nM T16347 C2L8DY 56679985 IC50 = 6000 nM T16347 C73OYR 56679986 IC50 = 2300 nM T16347 C5PM4N 56679987 IC50 = 6000 nM T16347 C2WDB7 56680468 Ki = 4000 nM T16347 CEK3S2 56680547 IC50 = 20900 nM T16347 CK1R7V 56681853 IC50 = 60100 nM T16347 C72JTU 56681854 IC50 = 8700 nM T16347 CJ50EL 56681855 IC50 = 6700 nM T16347 C05WLQ 56683006 IC50 = 14900 nM T16347 C4M6EC 56683323 IC50 = 9000 nM T16347 C6FEN9 56683324 IC50 = 33000 nM T16347 C1N9JZ 56683325 IC50 = 14000 nM T16347 C2MX8E 56683798 Ki = 5660 nM T16347 CN3EW7 56683882 IC50 = 15300 nM T16347 C5CQY2 56683883 IC50 = 26000 nM T16347 CV4PW2 56683884 Ki = 3900 nM T16347 CRVS72 56945877 IC50 = 100000 nM T16347 CJH0U3 56949846 IC50 = 9 nM T16347 C23KMR 56949985 IC50 = 11 nM T16347 C82OHP 56960992 IC50 = 900 nM T16347 CCS5X4 56961135 IC50 = 500 nM T16347 CI0Q1M 57327698 IC50 = 12140 nM T16347 CN5HO3 57327771 IC50 = 9240 nM T16347 CZP28F 57327772 IC50 = 4780 nM T16347 CO2F6B 57327843 IC50 = 7930 nM T16347 CIQP45 57327844 IC50 = 3660 nM T16347 C76UIC 57327845 IC50 = 2200 nM T16347 C1N9XS 57327846 Ki = 310 nM T16347 C79IOT 57327917 IC50 = 1350 nM T16347 CJYU43 57328789 IC50 = 13230 nM T16347 CT2X8K 57329174 IC50 = 2800 nM T16347 CWB63E 57345644 IC50 = 8300 nM T16347 CG71TE 57380427 IC50 > 10000000 nM T16347 C4QJD7 57380429 IC50 > 10000000 nM T16347 CLTX25 57380431 IC50 > 10000000 nM T16347 CU94DW 57380433 IC50 = 135000 nM T16347 CCY75L 57380662 IC50 > 10000000 nM T16347 CE24LJ 57380664 IC50 = 334000 nM T16347 CWZ9E2 57380666 IC50 > 10000000 nM T16347 C9H7GI 57380668 IC50 > 10000000 nM T16347 C25TFE 57390656 IC50 = 288 nM T16347 C70LDN 57390657 IC50 = 17 nM T16347 CXW05S 57390693 IC50 = 137000 nM T16347 CN5A1Q 57391733 IC50 = 1050 nM T16347 CW90NK 57391788 IC50 = 1200 nM T16347 CR2O3W 57392457 IC50 = 41 nM T16347 CR3Y5U 57393471 IC50 = 6200 nM T16347 C9OCN0 57393518 IC50 = 1300 nM T16347 CIM2X4 57394165 IC50 = 47 nM T16347 C6A7UF 57394166 IC50 = 480 nM T16347 C38BYE 57394167 IC50 = 38 nM T16347 CUT20F 57395175 IC50 > 50000 nM T16347 CE6W5J 57395192 IC50 = 1180 nM T16347 CL3O6H 57395194 IC50 = 2550 nM T16347 CZN24O 57395947 IC50 = 141 nM T16347 C9W0OB 57395948 IC50 = 31 nM T16347 CP8D0F 57395949 IC50 = 39 nM T16347 CE57HQ 57395972 IC50 = 6640 nM T16347 C56JAF 57396972 IC50 = 2030 nM T16347 C6WY1Q 57396974 IC50 = 940 nM T16347 CHEM09 57396976 IC50 = 1430 nM T16347 CQ6NK9 57397734 IC50 = 35 nM T16347 CN0RT3 57397735 IC50 = 500 nM T16347 CPO0R8 57397736 IC50 = 470 nM T16347 CGC16T 57397768 IC50 = 91700 nM T16347 C18FTX 57397769 IC50 = 217000 nM T16347 CQNG21 57397770 IC50 > 10000000 nM T16347 CKL3A8 57398721 IC50 = 950 nM T16347 C9VOI8 57398723 IC50 = 1690 nM T16347 CTV86F 57398725 IC50 = 3200 nM T16347 CT1GD4 57398727 IC50 = 3800 nM T16347 C1DG8N 57398729 IC50 = 3350 nM T16347 C3Q9DA 57398755 IC50 = 570 nM T16347 CK7YX1 57399401 IC50 = 35 nM T16347 CX3A5R 57399431 IC50 = 373000 nM T16347 CR32ZH 57400364 IC50 = 24500 nM T16347 C9G7RH 57400394 IC50 = 1150 nM T16347 CH0Y4N 57400437 IC50 = 5600 nM T16347 CF8QD0 57400441 IC50 = 1020 nM T16347 C2OK3M 57401165 IC50 = 18 nM T16347 CY27OL 57402190 IC50 = 1050 nM T16347 CL32MT 57402244 IC50 = 1410 nM T16347 C3C7UV 57402927 IC50 = 460 nM T16347 CME9A6 57403824 IC50 > 50000 nM T16347 CRW16Q 57403926 IC50 = 19700 nM T16347 CK7ND0 57404470 Ki = 800 nM T16347 C36GMW 57404471 Ki = 600 nM T16347 CVT2F6 57404472 Ki = 300 nM T16347 C1HJ0B 57404473 Ki = 400 nM T16347 COME35 57404494 Ki = 500 nM T16347 C9ZR5P 57404495 Ki = 500 nM T16347 CW0DR4 57408542 IC50 = 10400 nM T16347 CQ5DK4 57408657 IC50 = 2200 nM T16347 C1FSE5 57408658 IC50 = 5600 nM T16347 CBK1V0 57408659 Ki = 1200 nM T16347 CVN96U 57408660 IC50 = 2400 nM T16347 CX0AC6 57408661 IC50 = 10900 nM T16347 CFPD92 57408777 IC50 = 2500 nM T16347 C4E2UK 57408778 IC50 = 5100 nM T16347 CE8GS6 57408779 IC50 = 3000 nM T16347 C4L9EH 57408780 IC50 = 9000 nM T16347 CL7SH5 57456994 IC50 = 29800 nM T16347 CJ9AC8 57484282 IC50 = 270 nM T16347 CU5ND3 57514697 IC50 = 190000 nM T16347 C25GCF 57606999 IC50 = 1350 nM T16347 CYM68P 57607015 IC50 = 2430 nM T16347 C0HC3Q 57607021 IC50 = 1180 nM T16347 C3B4GV 57607023 IC50 = 960 nM T16347 C7Q2GB 57607037 IC50 = 430 nM T16347 C2OGL4 57607041 IC50 = 620 nM T16347 CWP53X 58021150 IC50 = 5600 nM T16347 CU2PT9 58537218 IC50 = 100000 nM T16347 COC4V3 58746455 IC50 = 2697739.43 nM T16347 C8LMQ6 58746458 IC50 = 1599558.03 nM T16347 CCV58M 58746466 IC50 = 339625.27 nM T16347 CC2A1W 58746519 IC50 = 179887.09 nM T16347 C3MB5I 58746527 IC50 = 1199499.3 nM T16347 C4LHX7 58746545 IC50 = 1499684.84 nM T16347 CUM87R 58746618 IC50 = 1000000 nM T16347 CD52ZT 58746630 IC50 = 169824.37 nM T16347 C1F3UW 58746662 IC50 = 1798870.92 nM T16347 CK2WG5 58746680 IC50 = 169824.37 nM T16347 CC34YL 58746703 IC50 = 790678.63 nM T16347 C7T9HR 58746729 IC50 = 1399587.32 nM T16347 C3JGM8 58746753 IC50 = 169824.37 nM T16347 CP10LO 58746871 IC50 = 5997910.76 nM T16347 CF71BW 59350289 IC50 = 12300 nM T16347 C4HTA7 59350381 IC50 > 20000 nM T16347 C0IQ7G 59439482 IC50 = 13000 nM T16347 COHJ70 59439485 IC50 = 23880 nM T16347 CKC0J6 59908232 IC50 = 17498.47 nM T16347 CYA1U7 60141123 IC50 = 10200 nM T16347 CH4U8X 60141550 IC50 = 10000 nM T16347 C4ZE0T 60142018 IC50 = 8300 nM T16347 COH1S4 60142154 IC50 = 8100 nM T16347 C49OYN 60142155 IC50 = 3200 nM T16347 CIZ45U 60148490 IC50 = 73200 nM T16347 CCS58F 60151889 IC50 = 3300 nM T16347 CS4Z8B 60151891 IC50 = 14000 nM T16347 C98DAR 60151894 IC50 = 155000 nM T16347 CY9C1B 60152033 IC50 = 11000 nM T16347 CZ41IL 60152037 IC50 = 172000 nM T16347 C2WQ3S 60152176 IC50 = 133000 nM T16347 C7YXQ6 60155758 IC50 = 6800 nM T16347 C5B7ES 60155759 IC50 = 6800 nM T16347 COPM73 60155760 IC50 = 6800 nM T16347 CYFU73 60155761 IC50 = 6800 nM T16347 CI81OU 60201376 IC50 = 27800 nM T16347 CD29BX 60201377 IC50 = 15200 nM T16347 CZ8ID6 66848959 IC50 = 300 nM T16347 CJ7AP3 67762287 IC50 = 510 nM T16347 C2M8NX 67859396 IC50 = 8800 nM T16347 CW2FZ3 68075819 IC50 = 4600 nM T16347 CSL3N8 68075861 IC50 = 4800 nM T16347 CPY5S8 68075863 IC50 = 5000 nM T16347 C92NMX 68122136 IC50 > 100000 nM T16347 CL18GV 70036097 Ki = 8800 nM T16347 C7BL9R 70036109 Ki = 15135.61 nM T16347 CP10SK 70240311 IC50 = 400 nM T16347 C2BT9H 70673568 IC50 = 10000 nM T16347 C2NRD9 70680338 IC50 = 18000 nM T16347 C4X1OZ 70681225 Ki = 1100 nM T16347 C0LU2D 70681226 Ki = 40000 nM T16347 C7T2VK 70682276 IC50 = 6800 nM T16347 C7K8VJ 70682727 IC50 = 15100 nM T16347 C9IRH5 70682728 IC50 = 1900 nM T16347 CRAM38 70683306 Ki = 7800 nM T16347 CW23BC 70683307 Ki = 1500 nM T16347 CHXY05 70684810 IC50 = 38400 nM T16347 CJQ31W 70684811 IC50 = 24800 nM T16347 C9WXM3 70684863 IC50 = 6300 nM T16347 CD76OS 70685412 Ki = 7800 nM T16347 CRJX90 70685413 Ki = 7700 nM T16347 CAM04W 70685414 Ki = 5100 nM T16347 CM5U9Y 70685415 Ki = 2400 nM T16347 C0K4UW 70685416 Ki = 1800 nM T16347 C1VT4H 70686947 IC50 > 100000 nM T16347 CV96RN 70686948 IC50 = 24500 nM T16347 C08RYT 70686949 IC50 > 100000 nM T16347 C0WO9M 70686969 IC50 = 2400 nM T16347 C6AG8L 70686970 IC50 = 1300 nM T16347 C5X7MP 70686971 IC50 = 1400 nM T16347 CQ1V4D 70686972 IC50 = 1300 nM T16347 CAZ01L 70687556 Ki = 1400 nM T16347 C37QPS 70688370 IC50 = 8800 nM T16347 C1ZD2P 70689036 IC50 > 100000 nM T16347 C03KXA 70689037 IC50 = 9600 nM T16347 C93VJQ 70689038 IC50 = 2500 nM T16347 C4NU1S 70689620 Ki = 1200 nM T16347 C1DN6B 70689621 Ki = 2900 nM T16347 CA64BK 70691129 IC50 > 100000 nM T16347 CRL18P 70691143 IC50 > 100000 nM T16347 CH5Z8E 70691144 IC50 > 100000 nM T16347 C8ORQ5 70691145 IC50 > 100000 nM T16347 CK3XG4 70691146 IC50 = 2600 nM T16347 CJ89TR 70691147 IC50 = 5100 nM T16347 CO6W0V 70691148 IC50 = 10400 nM T16347 CSF2C5 70693259 IC50 > 100000 nM T16347 CP37SW 70693260 IC50 = 22000 nM T16347 C16IZQ 70693261 IC50 = 5800 nM T16347 C49KWD 70693815 Ki = 4000 nM T16347 CBQ5X8 70695329 IC50 > 100000 nM T16347 C3HM8X 70695347 IC50 = 44400 nM T16347 CC1EV5 70695348 IC50 = 3300 nM T16347 CAI76J 70695349 IC50 = 9700 nM T16347 CKB7G3 70695350 IC50 = 2000 nM T16347 C2XP0G 70695935 Ki = 16300 nM T16347 CJY7W2 70697356 IC50 = 84600 nM T16347 CO24ET 70697357 IC50 = 8600 nM T16347 C6AX2Z 70697358 IC50 = 1500 nM T16347 CG56MJ 70697359 IC50 = 5000 nM T16347 CJ6IH4 70697438 IC50 = 17400 nM T16347 C3AJ7H 70981706 IC50 = 6700 nM T16347 CP4H6L 70981726 IC50 = 4500 nM T16347 C2KS7Y 70982811 IC50 = 5100 nM T16347 CJ48QM 71296672 IC50 = 15200 nM T16347 C7VES4 71449486 IC50 = 3560 nM T16347 CN0F5Z 71449491 IC50 = 7090 nM T16347 C4XUW1 71450557 IC50 = 39440 nM T16347 CHL47W 71450558 Ki = 840 nM T16347 CY1Z3K 71450598 IC50 = 20400 nM T16347 CD02LC 71450760 IC50 = 6710 nM T16347 C2TQY9 71451289 IC50 = 2050 nM T16347 C7EPN1 71451291 IC50 = 4890 nM T16347 COE35L 71452472 IC50 = 18600 nM T16347 CQ68KZ 71452583 IC50 > 60000 nM T16347 C3GAM4 71452584 IC50 = 7630 nM T16347 CGL2W9 71452585 IC50 = 5350 nM T16347 C21MPJ 71452586 IC50 = 5700 nM T16347 CY9H6K 71453112 IC50 = 4420 nM T16347 CR5E7G 71453113 IC50 = 3570 nM T16347 CBX20M 71453114 IC50 = 6300 nM T16347 CQB73X 71453167 IC50 = 550 nM T16347 CKV85O 71454347 IC50 = 4410 nM T16347 C2GBJ0 71454348 IC50 = 5230 nM T16347 CPRL17 71454955 IC50 = 4600 nM T16347 C7WUM1 71455905 IC50 > 40000 nM T16347 CPZ17Q 71456090 IC50 > 60000 nM T16347 C5XB2N 71456091 IC50 = 2800 nM T16347 CR84HE 71456092 IC50 = 3460 nM T16347 CY07HW 71456616 Ki = 700 nM T16347 CNW6F3 71457701 IC50 = 13200 nM T16347 C72UIR 71457702 IC50 = 28220 nM T16347 CW9OR3 71457703 IC50 = 9110 nM T16347 CX49EA 71457901 IC50 > 60000 nM T16347 CJU9C6 71457902 IC50 = 9820 nM T16347 CGZI63 71457903 IC50 = 4590 nM T16347 CXS4W0 71459613 IC50 = 11650 nM T16347 CXI25S 71459627 IC50 = 820 nM T16347 CXG3J6 71459672 IC50 = 19200 nM T16347 CM7W3N 71459673 IC50 = 12500 nM T16347 C6WL4I 71460322 IC50 = 2100 nM T16347 CPN94R 71460437 IC50 > 30000 nM T16347 C0FU8V 71461350 IC50 = 9270 nM T16347 CTY9V5 71461351 IC50 = 5570 nM T16347 CJOI01 71461352 IC50 = 19164 nM T16347 CAR47J 71461461 IC50 = 13900 nM T16347 CP43AS 71461531 IC50 = 2300 nM T16347 C25CKX 71462022 IC50 = 6370 nM T16347 C4Z0PS 71462023 IC50 = 2760 nM T16347 CQF79H 71462024 IC50 = 4950 nM T16347 C78NSM 71463071 IC50 = 9040 nM T16347 CQ5HR9 71463072 IC50 = 8620 nM T16347 CV76YL 71463073 IC50 = 3610 nM T16347 C0PO3Z 71463074 IC50 = 9130 nM T16347 C2VO3J 71463075 IC50 = 4110 nM T16347 C30MIG 71463268 IC50 = 3370 nM T16347 CUY43P 71463479 Ki = 30000 nM T16347 C6GIT7 71463480 Ki = 56000 nM T16347 CQ4FD7 71463481 Ki = 34000 nM T16347 C3I6MG 71463488 Ki = 25000 nM T16347 CV0ZA5 71467785 IC50 = 10600 nM T16347 C4N3CF 71496104 IC50 = 8660000 nM T16347 CWJ2O7 71496218 IC50 = 6830000 nM T16347 CTU0X5 71496219 IC50 = 6090000 nM T16347 CDPI81 71517216 IC50 = 23000 nM T16347 CWXP68 71517217 IC50 = 49000 nM T16347 C6LY3E 71517218 IC50 = 24500 nM T16347 CXI0F3 71561559 IC50 > 100000 nM T16347 CE0Y3O 71561685 IC50 = 14600 nM T16347 C3M4CF 71561686 IC50 = 12000 nM T16347 C82KCZ 71561687 IC50 = 6300 nM T16347 CDA8P2 71561688 IC50 > 30000 nM T16347 C87EXF 71561689 IC50 = 5200 nM T16347 CP9HX5 71561815 IC50 = 1200 nM T16347 C9H5YS 71561816 IC50 = 8000 nM T16347 C61MWP 71561817 IC50 = 12000 nM T16347 C9GO5M 71561818 IC50 = 60000 nM T16347 CWA30F 71561819 IC50 = 7400 nM T16347 CBC4G0 71561820 IC50 = 8400 nM T16347 CPV8Y3 71561944 IC50 = 8000 nM T16347 CCO57Q 71575995 Ki = 8900 nM T16347 C3C4PA 71578079 IC50 = 42500 nM T16347 CPN85Z 71578080 IC50 = 35200 nM T16347 C5D1TB 71592133 IC50 = 7000 nM T16347 CPWU40 71597177 IC50 > 50000 nM T16347 CPS6D0 71600596 Ki > 500000 nM T16347 CKV59P 71602348 Ki = 228000 nM T16347 C2U7LJ 71602401 Ki = 331000 nM T16347 CAT7J6 71602467 Ki = 211500 nM T16347 CM1P8W 71602468 Ki = 67500 nM T16347 CKA1R4 71602470 Ki = 125000 nM T16347 C28ILM 71602532 Ki = 66500 nM T16347 C1AB6Y 71602534 Ki = 82400 nM T16347 CR2SG8 71602535 Ki = 41000 nM T16347 CRM15H 71602536 Ki = 10000 nM T16347 CN7C8X 71602597 Ki = 162000 nM T16347 C0K4VR 71602598 Ki = 6800 nM T16347 C7BUG9 71602599 Ki = 35000 nM T16347 CQB81R 71602600 Ki = 7700 nM T16347 C5QO4E 71602654 Ki = 16800 nM T16347 CY82XN 71602655 Ki = 14900 nM T16347 CFH8Q1 71602656 Ki = 235000 nM T16347 CH2ON1 71602704 Ki = 14000 nM T16347 CQAZ96 71602705 Ki = 125000 nM T16347 CLC8M6 71602706 Ki = 82400 nM T16347 CW2J1C 71602708 Ki = 62000 nM T16347 C1B2KX 71602753 Ki = 68800 nM T16347 CB71UL 71602754 Ki = 92000 nM T16347 C0JW6B 71602804 Ki = 23600 nM T16347 C9Q7PN 71607898 IC50 = 2000 nM T16347 C2I7SU 71660814 IC50 = 7120 nM T16347 C5AHG6 71716739 IC50 = 13100 nM T16347 CC1RW5 71717335 IC50 = 8400 nM T16347 CT4MK9 71717989 IC50 > 50000 nM T16347 CPBR60 71718556 IC50 > 50000 nM T16347 C1P3VH 71718619 IC50 = 19500 nM T16347 CNA8L6 71719571 IC50 = 3600 nM T16347 CTQM06 71719757 IC50 > 50000 nM T16347 C2BL9Q 71719758 IC50 > 50000 nM T16347 CCY15D 71734765 IC50 = 1700 nM T16347 CRD9Y2 71770297 IC50 = 5950 nM T16347 CGC0E2 71770417 IC50 >= 20 ug.mL-1 T16347 C19RPW 71770419 IC50 >= 20 ug.mL-1 T16347 C5AG1C 72163286 IC50 = 33420 nM T16347 CTHK16 72163287 IC50 = 48180 nM T16347 CS0XU2 72163288 IC50 = 25620 nM T16347 C6F1TD 72163289 IC50 = 24880 nM T16347 C9R8ND 72163290 IC50 = 22560 nM T16347 C0FWS2 72163422 IC50 = 14830 nM T16347 C2RNH4 72163424 IC50 = 78190 nM T16347 CNLB62 72163425 IC50 = 35230 nM T16347 CT1G6F 72163427 IC50 = 24080 nM T16347 C6JMD4 72163430 IC50 = 29000 nM T16347 CB5M4P 72163577 IC50 = 27960 nM T16347 CE9VO5 72163579 IC50 = 22380 nM T16347 CUQ3P4 72163709 IC50 = 29680 nM T16347 CZJ80C 72163710 IC50 = 4540 nM T16347 CPKZ17 72163711 IC50 = 31420 nM T16347 CDO51E 72163712 IC50 = 44980 nM T16347 C94HFU 72165182 IC50 = 11010 nM T16347 CMC9L2 72190151 Ki = 680 nM T16347 CL70MO 72196940 IC50 = 1910 nM T16347 CYB36C 72196942 IC50 = 12200 nM T16347 CI67LN 72197305 IC50 = 9210 nM T16347 CULV83 72197478 IC50 = 16100 nM T16347 C63KSF 72545045 IC50 = 40300 nM T16347 C61PBV 72545046 IC50 = 10400 nM T16347 C0ZP1L 72545279 IC50 = 1300 nM T16347 C0RMO9 72947031 IC50 = 19560 nM T16347 CK07NR 73346398 IC50 = 8790 nM T16347 CCLA45 73347904 IC50 = 4420 nM T16347 C8LJ4Y 73347905 IC50 = 4880 nM T16347 CQEN46 73347906 IC50 = 5560 nM T16347 CKAP38 73347907 IC50 = 4180 nM T16347 CVU91E 73347908 IC50 = 1180 nM T16347 C90TVU 73348789 Ki = 6700 nM T16347 CR75AE 73348832 Ki = 63000 nM T16347 CEAS06 73349437 IC50 = 2680 nM T16347 C7RC5B 73349438 IC50 = 710 nM T16347 C8CR7H 73350368 Ki = 35000 nM T16347 CY0ER6 73350411 Ki = 18 nM T16347 C5X7UJ 73350460 IC50 = 2420 nM T16347 C0SMW4 73350687 IC50 >= 20 ug.mL-1 T16347 CUIC45 73350688 IC50 = 27200 nM T16347 CM1W6X 73352369 IC50 = 8300 nM T16347 C2T6FA 73352477 IC50 = 10550 nM T16347 CW1A0Y 73352478 IC50 = 770 nM T16347 C9Q8AJ 73352945 Ki = 170 nM T16347 CXL8I5 73353025 Ki = 200 nM T16347 CIDT03 73353949 IC50 = 8120 nM T16347 C5Z9MQ 73353950 IC50 = 6000 nM T16347 C3B4CD 73353951 IC50 = 3790 nM T16347 C1DWU4 73353952 IC50 = 1010 nM T16347 CSIZ58 73353953 IC50 = 2820 nM T16347 C9UP3V 73353954 IC50 = 540 nM T16347 CCH1Y6 73354070 IC50 = 52200 nM T16347 CRZ62F 73355036 IC50 = 1420 nM T16347 CS5O4J 73355491 IC50 = 1170 nM T16347 CJ67VI 73355492 IC50 = 2280 nM T16347 C92RWB 73355493 IC50 = 1620 nM T16347 C3KI2M 73355595 IC50 = 5000 nM T16347 C0V9NT 73356063 Ki = 18000 nM T16347 CMDC47 73357035 IC50 = 1420 nM T16347 CY0K7L 73357036 IC50 = 1120 nM T16347 C2YSV0 73357037 IC50 = 2560 nM T16347 C9J8IH 76308036 Ki = 93000 nM T16347 CY3XM0 76308037 Ki = 16982.44 nM T16347 CE7FT1 76308038 Ki = 74000 nM T16347 CC78MI 76308571 IC50 = 510 nM T16347 C36LWR 76308572 IC50 = 720 nM T16347 CKR8G5 76309919 IC50 > 30000 nM T16347 C7TOF4 76310031 IC50 = 9500 nM T16347 C2UMO6 76310032 IC50 = 24600 nM T16347 CL7JW5 76311652 Ki = 35000 nM T16347 C6MF1Y 76311979 Ki = 135000 nM T16347 C7PF2Z 76312236 IC50 = 2670 nM T16347 CD13GX 76312237 IC50 = 2720 nM T16347 CZX89S 76312238 IC50 = 520 nM T16347 C4PA7C 76312239 IC50 = 600 nM T16347 CFR39W 76312264 IC50 = 590 nM T16347 C46DLF 76312265 IC50 = 560 nM T16347 CT81WH 76312266 IC50 = 450 nM T16347 CL83ZG 76312267 IC50 = 3310 nM T16347 CP98WE 76313171 IC50 = 100000000 nM T16347 CBM2I6 76315206 Ki = 4700 nM T16347 C34MJU 76315207 Ki = 23988.33 nM T16347 CXN43S 76315784 IC50 = 550 nM T16347 C8ER9J 76315785 IC50 = 440 nM T16347 C68OQS 76315819 IC50 = 2100 nM T16347 CZJR13 76317135 IC50 > 30000 nM T16347 CF26QP 76317256 Ki = 500 nM T16347 C12KDX 76317257 Ki = 1500 nM T16347 CFR42O 76318860 Ki = 3388.44 nM T16347 CW3N7T 76318861 Ki = 13800 nM T16347 C8C0BU 76318897 Ki = 16982.44 nM T16347 CK48HJ 76319196 Ki = 63000 nM T16347 CHN3Z5 76319197 Ki = 48000 nM T16347 CCN40D 76319472 IC50 = 660 nM T16347 CY8R9M 76319473 IC50 = 590 nM T16347 CU57ZO 76319507 IC50 = 4620 nM T16347 CJS2E1 76319508 IC50 = 610 nM T16347 CT6W0M 76319509 IC50 = 880 nM T16347 CJI8Y2 76319510 IC50 = 780 nM T16347 C3LYQ7 76320443 IC50 = 100000000 nM T16347 CELQ61 76320957 IC50 = 3900 nM T16347 C2L0IY 76320960 IC50 = 4000 nM T16347 C64OWT 76322515 Ki = 1200 nM T16347 CYK3S1 76322853 Ki = 150000 nM T16347 C72OTI 76323095 IC50 = 150 nM T16347 CJ9RZ6 76323096 IC50 = 630 nM T16347 CB1P7M 76323097 IC50 = 530 nM T16347 C8TR0Z 76323125 IC50 = 570 nM T16347 C85LPV 76324628 IC50 = 7500 nM T16347 C1FNK8 76324629 IC50 = 4600 nM T16347 CTI5H1 76326107 Ki = 60000 nM T16347 C7J1FT 76326418 Ki = 170000 nM T16347 CQ78WV 76326683 IC50 = 550 nM T16347 C78VFN 76327608 IC50 = 14996848.36 nM T16347 C5NEJ8 76327640 IC50 = 69984199.6 nM T16347 C6QJV8 76328065 IC50 > 30000 nM T16347 C7LS8E 76328072 IC50 = 23900 nM T16347 CZ9C5F 76328193 IC50 = 2200 nM T16347 C59MCI 76329706 Ki = 1700 nM T16347 CC1DR4 76329744 Ki = 23988.33 nM T16347 C2W8QX 76329745 Ki = 10964.78 nM T16347 CAJ97D 76329746 Ki = 14000 nM T16347 CZ9IT4 76330041 Ki = 48000 nM T16347 C9B5RE 76330317 IC50 = 820 nM T16347 CF0AD2 76330318 IC50 = 650 nM T16347 CFS5L6 76330347 IC50 = 1330 nM T16347 CXWO63 76330348 IC50 = 16350.01 nM T16347 C3IT0A 76331872 Ki = 1500 nM T16347 C0K9JN 76331873 IC50 = 1600 nM T16347 CIAH20 76331876 IC50 = 1100 nM T16347 CJ0D8G 76333370 Ki = 1288.25 nM T16347 CVU26L 76333371 Ki = 38904.51 nM T16347 CB5IG2 76333407 Ki = 1800 nM T16347 CX7KO4 76333950 IC50 = 570 nM T16347 C5EP0S 76335338 IC50 = 3900 nM T16347 C2HG0O 76335442 Ki = 2300 nM T16347 CWM07I 77461140 IC50 = 2340 nM T16347 CB2ZT4 78318903 IC50 = 26980 nM T16347 C60WKI 85587091 Ki = 19940 nM T16347 CYI4X8 86302286 IC50 = 6440 nM T16347 CC2Z4G 86302611 IC50 = 9710 nM T16347 C6RZ5H 86302612 IC50 = 9970 nM T16347 CBY97E 86766296 IC50 = 16540 nM T16347 CT1JH8 86766297 IC50 = 9500 nM T16347 CFZ0E8 86766298 IC50 = 5040 nM T16347 C60NUB 86766299 IC50 = 2650 nM T16347 C0I9VX 86766300 IC50 = 14630 nM T16347 CJL4M8 86766301 IC50 = 12160 nM T16347 CYA7X6 86766302 IC50 = 10240 nM T16347 CR4DW5 86766303 IC50 = 4610 nM T16347 CNF6D8 86766304 IC50 = 11050 nM T16347 CA4LO9 86766305 IC50 = 5370 nM T16347 CL4IN3 86766306 IC50 = 5960 nM T16347 C6NL3Q 86766307 IC50 = 7140 nM T16347 CGML73 86766308 IC50 = 26540 nM T16347 CECP92 90643583 IC50 = 378000 nM T16347 CZ39XP 90643584 IC50 = 716500 nM T16347 C0WLO3 90645362 IC50 < 10000 nM T16347 CB7ZI8 90645363 IC50 < 10000 nM T16347 CQ9MI1 90645364 IC50 < 10000 nM T16347 CG0M4L 90645365 IC50 < 10000 nM T16347 CU6CS4 90645366 IC50 < 10000 nM T16347 CSC73N 90645367 IC50 < 10000 nM T16347 CR4UE0 90645368 IC50 < 10000 nM T16347 CH6KI0 90645369 IC50 < 10000 nM T16347 C2N7QU 90645370 IC50 < 10000 nM T16347 CHO32F 90645371 IC50 < 10000 nM T16347 CE1X3F 90645372 IC50 < 10000 nM T16347 CJ4DB7 90645373 IC50 < 10000 nM T16347 CH1ZF7 90645374 IC50 < 10000 nM T16347 CQO89G 90645375 IC50 < 10000 nM T16347 CF2M1A 90645376 IC50 < 10000 nM T16347 CO94JV 90645377 IC50 < 10000 nM T16347 C4DR1Z 90645378 IC50 < 10000 nM T16347 C9VAM1 90645379 IC50 < 10000 nM T16347 CD71LB 90645380 IC50 < 10000 nM T16347 CW4G8S 90645381 IC50 < 10000 nM T16347 CI0XF1 90654915 IC50 = 17230 nM T16347 C5LN3W 90654916 IC50 = 15870 nM T16347 C52OZB 90654917 IC50 = 6530 nM T16347 CBZ54P 90654918 IC50 = 16560 nM T16347 CI72XV 90654919 IC50 = 5670 nM T16347 CDYZ58 90654920 IC50 = 26490 nM T16347 CY16IS 90654921 IC50 = 10360 nM T16347 C3MXR1 90654922 IC50 = 1030 nM T16347 CQU90K 90654923 IC50 = 780 nM T16347 C6MQ9U 90654924 IC50 = 3120 nM T16347 C32TGW 90654925 IC50 = 20370 nM T16347 CCH19N 90666310 IC50 = 16090 nM T16347 C7H1VW 90666311 IC50 = 11370 nM T16347 C1GVI3 90666312 IC50 > 40000 nM T16347 C0C5HY 90666313 IC50 > 40000 nM T16347 CG26AC 90666314 IC50 > 40000 nM T16347 C8GV2N 90666315 IC50 > 40000 nM T16347 C3SF8U 90666316 IC50 = 12390 nM T16347 CP94DI 90666344 IC50 = 1000 nM T16347 COLU57 90666450 IC50 = 15860 nM T16347 C2KV5C 90666451 IC50 = 7100 nM T16347 CS6ZL4 90666452 IC50 = 12480 nM T16347 CA7S4L 90666453 IC50 = 9660 nM T16347 CQTD23 90666454 IC50 = 5601 nM T16347 CBK96X 90666455 IC50 = 1600 nM T16347 C61PBQ 90666456 IC50 = 2080 nM T16347 C40WCO 90666457 IC50 = 3010 nM T16347 C2ZGE9 90666458 IC50 = 5940 nM T16347 CG5TY1 90666459 IC50 = 3680 nM T16347 CWQN87 90666460 IC50 = 5430 nM T16347 CLU52N 90666461 IC50 = 2320 nM T16347 C0DW7A 90666462 IC50 = 3050 nM T16347 CXMC74 90666463 IC50 = 2450 nM T16347 C92NVK 90666464 IC50 = 4420 nM T16347 C41BKW 90666808 IC50 = 7600 nM T16347 C6LE3C 90666812 IC50 = 7470 nM T16347 CAOY85 90666813 IC50 = 9910 nM T16347 C9FM7A 90666817 IC50 = 8060 nM T16347 C2ZA6I 90667494 IC50 = 88000 nM T16347 C2EXC3 97686398 IC50 = 49400 nM T16347 CUG92M 101022947 IC50 = 49400 nM T16347 C5Y0MH 101280188 IC50 = 8600 nM T16347 CC17JA 101565497 IC50 = 8500 nM T16347 C9HJ1X 101600045 IC50 = 2560 nM T16347 CTE61M 101681084 IC50 = 26800 nM T16347 C2E7SL 101681085 IC50 = 45200 nM T16347 CLVX03 101876538 IC50 = 24460 nM T16347 C26FMV 101876539 IC50 = 3140 nM T16347 C19JKD 101884098 IC50 = 65000 nM T16347 CLMR71 101886901 IC50 = 3800 nM T16347 CB4F7N 101910192 Ki = 10300 nM T16347 C1UJD8 102004659 Ki = 22900 nM T16347 CCI47Z 102036608 IC50 = 67100 nM T16347 C9K6GH 102194063 IC50 = 14900 nM T16347 CI1L0S 102194704 IC50 = 1340 nM T16347 CYW80L 102307785 IC50 = 170 nM T16347 C06GAQ 102331593 IC50 = 8200 nM T16347 C7K5UE 102519726 IC50 = 25200 nM T16347 CXPD14 118706083 IC50 = 20000 nM T16347 CI4XC1 118706086 IC50 = 7.5 ug.mL-1 T16347 C0CSP4 118706087 IC50 = 12.3 ug.mL-1 T16347 CF4B6Q 118706088 IC50 = 9.2 ug.mL-1 T16347 C9YQ6S 118706089 IC50 = 11.4 ug.mL-1 T16347 C7EWB3 118706090 IC50 = 14 ug.mL-1 T16347 CJ73OD 118706095 IC50 = 13.9 ug.mL-1 T16347 C74EMW 118706098 IC50 > 20 ug.mL-1 T16347 CM0LS8 118706099 IC50 = 8.1 ug.mL-1 T16347 CX9K8W 118706100 IC50 > 20 ug.mL-1 T16347 CX81PZ 118706101 IC50 = 3.1 ug.mL-1 T16347 CV5Q8J 118706102 IC50 = 2.4 ug.mL-1 T16347 CRP3V4 118706103 IC50 = 9.4 ug.mL-1 T16347 C89BPJ 118706104 IC50 = 6.5 ug.mL-1 T16347 CW23YS 118706105 IC50 = 45.2 ug.mL-1 T16347 CGOE34 118706499 IC50 = 11300 nM T16347 CFVG50 118706500 IC50 = 14200 nM T16347 C1ZR2S 118706501 IC50 = 8100 nM T16347 CO3Y8U 118706502 IC50 = 5300 nM T16347 C5JFV4 118706503 IC50 = 4900 nM T16347 C65FDN 118706504 IC50 = 7600 nM T16347 C2VT6G 118706505 IC50 = 22300 nM T16347 CAI73P 118706506 IC50 = 8100 nM T16347 CPU85N 118706507 IC50 = 8200 nM T16347 CN84ZO 118706508 IC50 = 17000 nM T16347 C1SD4T 118706509 IC50 = 4600 nM T16347 CN27VR 118706510 IC50 = 12300 nM T16347 C61MAP 118706511 IC50 = 10000 nM T16347 CY5X2U 118706512 IC50 = 10300 nM T16347 CT39ZX 118706513 IC50 = 12100 nM T16347 CGQ9U7 118706514 IC50 = 7900 nM T16347 C6LIY1 118706515 IC50 = 9700 nM T16347 CM1UT0 118706516 IC50 > 30000 nM T16347 C19HMC 118706517 IC50 = 6600 nM T16347 C8LB0S 118706518 IC50 = 12200 nM T16347 CTRP72 118706519 IC50 > 30000 nM T16347 CI2CB4 118706520 IC50 > 30000 nM T16347 CS2J9F 118706521 IC50 > 30000 nM T16347 CW6MN5 118706522 IC50 = 22700 nM T16347 CBN06F 118706523 IC50 = 20600 nM T16347 C7P3CA 118706524 IC50 > 30000 nM T16347 C20HQT 118706525 IC50 > 30000 nM T16347 C45ZYK 118706526 IC50 = 6400 nM T16347 CI67EM 118706527 IC50 > 30000 nM T16347 C2GS6K 118706852 IC50 = 12000 nM T16347 CEG3J5 118706853 IC50 = 9600 nM T16347 CDH5G7 118706854 IC50 = 7200 nM T16347 CX6C0I 118706855 IC50 = 29300 nM T16347 C3I9LQ 118708255 IC50 = 6430 nM T16347 CQ2T8J 118708258 IC50 = 6540 nM T16347 C3E2WA 118708261 IC50 = 7320 nM T16347 CRED83 118708263 IC50 = 7120 nM T16347 C0WNF2 118710330 IC50 = 4.07 ug.mL-1 T16347 CY8D7B 118710331 IC50 = 3.48 ug.mL-1 T16347 C25JPT 118710332 IC50 = 8.26 ug.mL-1 T16347 CU47TG 118710333 IC50 = 5.88 ug.mL-1 T16347 CH8TQ0 118710335 IC50 = 4.14 ug.mL-1 T16347 CM2Y3B 118710336 IC50 = 6.24 ug.mL-1 T16347 CFT67U 118710337 IC50 = 7.47 ug.mL-1 T16347 CIH1B8 118710339 IC50 = 8.75 ug.mL-1 T16347 CC3J7Q 118710340 IC50 = 4.25 ug.mL-1 T16347 C5PCY1 118710341 IC50 = 0.85 ug.mL-1 T16347 CQ1TN4 118710342 IC50 = 1.67 ug.mL-1 T16347 C7ZLK3 118710343 IC50 = 4.63 ug.mL-1 T16347 C47QMJ 118710344 IC50 = 4.2 ug.mL-1 T16347 CY6H1O 118710345 IC50 = 5.44 ug.mL-1 T16347 CN2XA6 118710346 IC50 = 3.63 ug.mL-1 T16347 CX89NJ 118710347 IC50 = 4.03 ug.mL-1 T16347 CUG17X 118710348 IC50 = 5.14 ug.mL-1 T16347 C7IOM9 118710349 IC50 = 1.88 ug.mL-1 T16347 CH38YV 118710350 IC50 = 5.33 ug.mL-1 T16347 CET9Z2 118710351 IC50 = 3.75 ug.mL-1 T16347 C87BLJ 118710352 IC50 = 2.9 ug.mL-1 T16347 CJUM81 118710353 IC50 = 3.34 ug.mL-1 T16347 CPJ98Q 118710355 IC50 = 1.69 ug.mL-1 T16347 CPS0R7 118710356 IC50 = 4.13 ug.mL-1 T16347 CP5NK7 118710357 IC50 = 1.36 ug.mL-1 T16347 CIQ1S5 118710358 IC50 = 8.04 ug.mL-1 T16347 CUD6A9 118710359 IC50 = 1.96 ug.mL-1 T16347 C9SH1O 118710360 IC50 = 3.2 ug.mL-1 T16347 CD7X4J 118716810 IC50 = 17800 nM T16347 CK69NP 118716811 Ki = 2100 nM T16347 CIV9Z7 118716812 Ki = 4800 nM T16347 CUY04G 118716813 IC50 = 36500 nM T16347 C36KIZ 118721518 IC50 = 2300 nM T16347 CM69SO 118721519 IC50 = 11010 nM T16347 CX2A8G 118722143 IC50 > 120000 nM T16347 CV5F0I 118722144 IC50 > 120000 nM T16347 CQ79XG 118725536 IC50 = 7450 nM T16347 CZ7GA5 118726285 Ki = 15100 nM T16347 C9FDH8 118726286 IC50 = 700 nM T16347 C0MYG1 118727014 IC50 > 40000 nM T16347 C8JB4K 118727015 IC50 > 40000 nM T16347 CQGO51 118727016 IC50 > 35000 nM T16347 C1PVK8 118727017 IC50 > 40000 nM T16347 CI3Z0W 118727934 Ki = 20050 nM T16347 C32ODE 118729111 IC50 = 6550 nM T16347 CTV62N 118729112 IC50 = 26350 nM T16347 CP9E4Q 118729113 IC50 = 23460 nM T16347 CS2XI7 118729114 IC50 = 4430 nM T16347 C3LN4T 118729115 IC50 = 5180 nM T16347 CF9KD7 118729116 IC50 = 4680 nM T16347 C27YKT 118729117 IC50 = 9120 nM T16347 C5FXC0 118729118 IC50 = 9700 nM T16347 C90UMX 118729119 IC50 = 10120 nM T16347 C0YGL1 118729120 IC50 = 590 nM T16347 CGTJ18 118729121 IC50 = 4270 nM T16347 C9LP2D 118729122 IC50 = 7260 nM T16347 C5D0SM 118729124 IC50 = 8850 nM T16347 C5GM1D 118729125 IC50 = 2680 nM T16347 CHF7U0 118729126 IC50 = 2730 nM T16347 CSI5O7 118729165 IC50 = 0.82 ug.mL-1 T16347 C4TY2N 118729167 IC50 = 4.42 ug.mL-1 T16347 C8S3ZX 118729169 IC50 = 9.59 ug.mL-1 T16347 C0IJ2X 118737463 IC50 = 12800 nM T16347 CRA4F3 118737464 Ki = 390 nM T16347 C4YS5W 118737466 Ki = 410 nM T16347 CI65JN 118737609 IC50 = 500 nM T16347 C82KRX 118737610 IC50 = 8200 nM T16347 CC2ZT6 118737611 IC50 = 5600 nM T16347 CY6K0I 118737612 IC50 = 15600 nM T16347 CB0CS9 118737613 IC50 = 600 nM T16347 CE4RH2 118737614 IC50 = 800 nM T16347 CA1VM7 118737695 IC50 = 1100 nM T16347 CU6SD1 118737696 IC50 = 800 nM T16347 CS93FJ 122178946 IC50 = 11300 nM T16347 C05ESG 122178947 IC50 > 30000 nM T16347 CN94HY 122178948 IC50 > 30000 nM T16347 C4Y7WE 122178949 IC50 > 30000 nM T16347 C9V4LR 122178950 IC50 = 4700 nM T16347 CC69NY 122179688 IC50 = 690 nM T16347 CH6OW5 122179777 IC50 = 13200 nM T16347 C19XDF 122179778 IC50 = 9800 nM T16347 CH0P4X 122180314 IC50 > 23000 nM T16347 CKY20N 122180315 IC50 > 23000 nM T16347 CDOV73 122180316 IC50 > 23000 nM T16347 CFQ6P8 122182191 IC50 = 537 nM T16347 CFUC86 122182192 IC50 = 309 nM T16347 CN02HB 122182193 IC50 = 212 nM T16347 CI87OL 122182194 IC50 = 203 nM T16347 CSP7V2 122182195 IC50 = 2733 nM T16347 C7UM1C 122182196 IC50 = 204 nM T16347 C51ZYN 122182197 IC50 = 756 nM T16347 CLB2T6 122184713 IC50 = 8400 nM T16347 CV9DR8 122186983 IC50 = 8700 nM T16347 CA1OU0 122186984 IC50 = 8500 nM T16347 CS4KV9 122186985 IC50 = 11900 nM T16347 C12OHP 122187565 IC50 = 9300 nM T16347 CXHR32 122187566 IC50 = 3000 nM T16347 C59OUG 122187567 IC50 = 7000 nM T16347 CC8ZT6 122193411 IC50 = 3500 nM T16347 C7H6UG 122193475 IC50 = 7400 nM T16347 C6M9PN 122193476 IC50 = 6600 nM T16347 C6QW0O 122193477 IC50 = 4100 nM T16347 CGNA34 122193478 IC50 = 10000 nM T16347 CRN54A 122193479 IC50 = 1300 nM T16347 CO37CZ 122193480 IC50 = 570 nM T16347 C5QUH9 122193481 IC50 = 3400 nM T16347 CLA24K 122193482 IC50 = 136000 nM T16347 C3OJ9A 122193483 IC50 = 8100 nM T16347 CMXE37 122193484 IC50 = 6800 nM T16347 C7ADN4 122193485 IC50 = 114000 nM T16347 CN74GH 122193486 IC50 = 110000 nM T16347 C0CV5O 122193487 IC50 = 960 nM T16347 CE5OT2 122193538 IC50 = 9700 nM T16347 CX8B2A 122193539 IC50 = 5100 nM T16347 CYV54X 122193540 IC50 = 11000 nM T16347 CX0U3Z 122193541 IC50 = 103000 nM T16347 CF2QP8 122193542 IC50 = 122000 nM T16347 CP47VC 122193543 IC50 = 113000 nM T16347 CO20ZD 122193544 IC50 = 89000 nM T16347 CQ5SU4 122193545 IC50 = 103000 nM T16347 CV5WA6 122193546 IC50 = 96000 nM T16347 C85LKT 122193547 IC50 = 142000 nM T16347 CI7WX9 122193548 IC50 = 104000 nM T16347 CMB90J 122193549 IC50 = 5400 nM T16347 C8Z0CD 122193550 IC50 = 101000 nM T16347 CH27TJ 122193551 IC50 = 22000 nM T16347 CJ6RO8 122193596 IC50 > 10000 nM T16347 C6KR0D 122194839 Ki = 1830 nM T16347 C85FQM 122194840 IC50 = 6100 nM T16347 C6SIU3 122194841 IC50 = 1700 nM T16347 CX2Y3K 122195056 IC50 = 2300 nM T16347 CR6P8H 122195057 IC50 = 2400 nM T16347 CQZ0J3 122195058 Ki = 4100000 nM T16347 CTK19P 122196239 IC50 = 16098 nM T16347 C5LEY0 122196240 IC50 = 346 nM T16347 CKT67D 122196241 IC50 = 222 nM T16347 CK35PR 122196242 IC50 = 902 nM T16347 CSB9Q4 122196243 IC50 = 896 nM T16347 C6Y4RQ 122196286 IC50 = 20338 nM T16347 C2PVC5 122196288 IC50 = 492 nM T16347 CV2H8T 122196290 IC50 = 470 nM T16347 CX6D7P 122196291 IC50 = 1709 nM T16347 CU3RP8 124141953 IC50 > 80000 nM T16347 CDBY61 124922745 IC50 = 63800 nM T16347 C46PST 127024952 IC50 = 9660 nM T16347 CF05SB 127025572 IC50 > 120000 nM T16347 C0KDZ2 127025573 IC50 = 13140 nM T16347 CI0NR9 127025574 IC50 = 12510 nM T16347 C6RI3J 127025575 IC50 = 8960 nM T16347 C5Z4PH 127025576 IC50 = 17260 nM T16347 C94EIF 127025577 IC50 = 13730 nM T16347 CR87HW 127025578 IC50 > 120000 nM T16347 CM9CP5 127027398 IC50 = 14060 nM T16347 C2A4GS 127027399 IC50 = 19720 nM T16347 CYOQ30 127027703 IC50 = 21930 nM T16347 CX52UN 127027704 IC50 = 24440 nM T16347 C6TIJ1 127027705 IC50 = 15780 nM T16347 C6H9SE 127027706 IC50 > 120000 nM T16347 C2X4JK 127027707 IC50 = 8800 nM T16347 C6UR4C 127027724 IC50 > 120000 nM T16347 C0RQ1U 127027725 IC50 = 16820 nM T16347 C0K2UI 127028022 IC50 = 15900 nM T16347 C1WA5T 127028346 IC50 = 18360 nM T16347 CC8HW0 127028347 IC50 > 120000 nM T16347 C6T0DY 127028683 IC50 = 26120 nM T16347 CL6QV7 127028684 IC50 = 21670 nM T16347 CG68NT 127028685 IC50 = 9660 nM T16347 C3MCH5 127028686 IC50 = 31490 nM T16347 C58GAU 127030486 IC50 = 6300 nM T16347 C76XUY 127030488 IC50 = 6800 nM T16347 CNGW74 127030567 IC50 = 7800 nM T16347 C6L8GA 127031122 IC50 = 7000 nM T16347 C8IEQ9 127031582 IC50 = 7500 nM T16347 CQ9R6U 127036995 Ki = 12300 nM T16347 CJ76FX 127037140 Ki = 3400 nM T16347 CK8IB2 127039596 IC50 = 64 nM T16347 CW9JQ8 127042510 IC50 = 1900 nM T16347 C0TP9X 127050084 IC50 = 936 nM T16347 CIAX67 127050086 IC50 = 50 nM T16347 C4WR2Y 127050690 IC50 = 7700 nM T16347 CK98DU 127050691 Ki = 170 nM T16347 CKPG08 127050931 IC50 = 1500 nM T16347 CWGC50 127051219 Ki = 4.9 nM T16347 CH1Y7Z 127051220 IC50 = 9600 nM T16347 CEL9C4 127052247 IC50 = 355 nM T16347 CXC3M0 127052248 IC50 = 16008 nM T16347 C7VW9K 127052249 IC50 = 4830 nM T16347 CEH0A6 132495287 Ki = 4600 nM T16347 CY4LI6 132495288 Ki = 4500 nM T16347 CD0UT1 132499765 IC50 = 450 nM T16347 C20SHK 132499766 IC50 = 1600 nM T16347 CLJE51 132499769 IC50 = 420 nM T16347 CRXG27 132499770 IC50 = 2700 nM T16347 C06DVG 132520250 IC50 = 3440 nM T16347 CF4U0D 132520252 IC50 = 6270 nM T16347 CG3QU6 132520254 IC50 = 7670 nM T16347 C7N5WD 132525259 IC50 = 6500 nM T16347 COVA15 132566461 IC50 = 1300 nM T16347 CO3K6Z 132566462 IC50 = 4300 nM T16347 C4SV0N 132566463 IC50 = 4300 nM T16347 C8LZ3N 132566465 IC50 = 4100 nM T16347 CP81IW 132566466 IC50 = 1800 nM T16347 CG2FU0 132566467 IC50 = 3000 nM T16347 CM3E9C 132566468 IC50 = 1600 nM T16347 CICG27 132852946 IC50 = 41000 nM T16347 C40HRA 132852953 IC50 = 52000 nM T16347 CF5HN6 132938289 IC50 = 13700 nM T16347 CO8V1Q 134130829 IC50 > 20000 nM T16347 CLS1B9 134131632 IC50 > 100000 nM T16347 C9BH3S 134131790 IC50 = 260400 nM T16347 C3Q6HX 134132029 IC50 > 20000 nM T16347 COG29Y 134132248 IC50 = 13800 nM T16347 C09GOE 134132259 IC50 = 23000 nM T16347 C2AX0E 134132301 IC50 = 10000 nM T16347 CXM14Y 134132344 IC50 > 20000 nM T16347 CN2R3H 134132944 IC50 = 4500 nM T16347 COB83U 134132961 IC50 = 6400 nM T16347 CY4N3A 134132971 IC50 > 20000 nM T16347 CJV5H9 134133280 IC50 = 17200 nM T16347 CQV2R8 134133435 IC50 = 14700 nM T16347 CAL9T7 134133803 IC50 = 14000 nM T16347 CIM15P 134134309 IC50 > 500000 nM T16347 CB73HC 134135216 IC50 = 24000 nM T16347 C9RLU5 134135241 IC50 = 7500 nM T16347 CY6X7Q 134135441 Ki = 8100 nM T16347 CLK4N7 134135565 IC50 = 37000 nM T16347 CV60GU 134135926 IC50 = 16000 nM T16347 C09YNW 134136545 IC50 = 11000 nM T16347 C8O2VJ 134136588 IC50 = 36000 nM T16347 C3SJ8A 134136833 Ki = 4400 nM T16347 CT2U6A 134136885 IC50 > 100000 nM T16347 CX4M9U 134137212 Ki = 4100 nM T16347 C97SXD 134137530 IC50 = 13000 nM T16347 CK1ED4 134137535 IC50 > 20000 nM T16347 CW3D7Y 134138036 IC50 = 37000 nM T16347 C0ETZ2 134138476 IC50 = 2900 nM T16347 C14VBN 134138533 IC50 = 3200 nM T16347 CO69VN 134138834 IC50 > 500000 nM T16347 CI5RT7 134138997 IC50 = 17000 nM T16347 C8ZBV3 134139324 IC50 = 23000 nM T16347 C9WV1I 134139428 IC50 > 20000 nM T16347 CI8UM3 134140100 IC50 = 36000 nM T16347 CCS63E 134140312 IC50 > 20000 nM T16347 CD6W2L 134140483 IC50 = 18000 nM T16347 C9YRW5 134140561 IC50 > 100000 nM T16347 CK23UB 134140778 IC50 = 6300 nM T16347 C4E0RK 134141025 Ki = 11000 nM T16347 CFVU60 134141414 IC50 > 20000 nM T16347 CWD9J0 134141423 IC50 = 14000 nM T16347 CW69FM 134143209 IC50 = 27000 nM T16347 C68CAL 134143448 IC50 = 56000 nM T16347 CPW0G8 134143816 IC50 > 100000 nM T16347 CJCA63 134143988 IC50 = 7000 nM T16347 CV3LS4 134144001 IC50 = 11000 nM T16347 CL05EQ 134144945 IC50 = 34000 nM T16347 C28JSW 134145140 IC50 = 27000 nM T16347 CZ7F2I 134146104 IC50 = 14000 nM T16347 C8BC1Z 134146721 IC50 = 27000 nM T16347 CQN18H 134147028 IC50 = 12000 nM T16347 C90HIR 134147609 Ki = 13000 nM T16347 C39WJL 134147836 IC50 = 14000 nM T16347 CJQ4M5 134148016 IC50 = 34000 nM T16347 C4E0TR 134148396 IC50 > 20000 nM T16347 C9NU1K 134148434 IC50 = 422400 nM T16347 CQ39KF 134148924 IC50 = 38000 nM T16347 CHW3T2 134149588 IC50 > 100000 nM T16347 CAVO70 134149830 IC50 = 28000 nM T16347 CRG1A0 134150611 IC50 > 20000 nM T16347 CI9C7J 134151413 IC50 = 9400 nM T16347 CV3CF6 134151444 IC50 = 12000 nM T16347 CR72FZ 134152023 IC50 > 20000 nM T16347 C8NY5U 134152045 IC50 = 8100 nM T16347 CC8FU2 134152403 IC50 > 100000 nM T16347 C1FGJ5 134152452 IC50 = 12600 nM T16347 CUTE29 134152660 IC50 = 11000 nM T16347 C72XBK 134152859 IC50 = 31000 nM T16347 C10YSH 134152958 IC50 = 8000 nM T16347 CBWE06 134153308 IC50 = 12000 nM T16347 CO24SI 134154614 IC50 > 20000 nM T16347 C56HZR 134154787 Ki = 8600 nM T16347 CJ7AE3 134155165 IC50 = 10000 nM T16347 CA2GM0 134155503 Ki = 7100 nM T16347 CQ5BU3 134156236 IC50 = 27000 nM T16347 CVW36N 134157472 IC50 = 16000 nM T16347 C5CU3J 134157618 IC50 > 20000 nM T16347 C7AT5S 134157744 IC50 = 24000 nM T16347 CN23HD 134157879 IC50 = 6600 nM T16347 C2V7NL 135797380 IC50 > 100000 nM T16347 C27EYJ 135797381 IC50 > 100000 nM T16347 CZOL36 135797386 IC50 > 100000 nM T16347 CBX75S 135797387 IC50 > 100000 nM T16347 C2L6UZ 135797388 IC50 > 100000 nM T16347 C0S1VO 135797389 IC50 > 100000 nM T16347 CS40TI 135797392 IC50 > 100000 nM T16347 C0RJW6 135797397 IC50 = 68100 nM T16347 CZC42X 135924009 IC50 = 9300 nM T16347 C5BL1Z 135924010 IC50 = 156600 nM T16347 C9UA3N 135924011 IC50 = 11300 nM T16347 C1V8JE 135924012 IC50 = 2500 nM T16347 C8HP1O 135924013 IC50 = 18800 nM T16347 CHUD85 135924014 IC50 = 7500 nM T16347 CTZ5K1 135924015 IC50 = 19400 nM T16347 CAF8B6 135924016 IC50 = 25700 nM T16347 CK4X8S 135924017 IC50 = 11400 nM T16347 CE1FB0 135924018 IC50 = 54900 nM T16347 C39EPD 135924019 IC50 = 32800 nM T16347 CEH2M5 135924020 IC50 = 63100 nM T16347 CN6I5O 135924021 IC50 = 38200 nM T16347 CKW8X5 135924023 IC50 > 300000 nM T16347 CO3EX1 135924024 IC50 = 37100 nM T16347 CBJ7F8 135924025 IC50 = 9800 nM T16347 C81SHP 135924026 IC50 = 15400 nM T16347 CI62JU 135924027 IC50 = 11700 nM T16347 CAL83P 135924028 IC50 = 14500 nM T16347 CJ14VX 135924029 IC50 = 19300 nM T16347 C5C4EP 135924030 IC50 = 1500 nM T16347 C5UL0V 135955126 IC50 > 100000 nM T16347 C85VGD 136069445 IC50 > 100000 nM T16347 C7MFW0 136088968 IC50 = 27630 nM T16347 C57SCL 136114690 IC50 = 460000 nM T16347 C42NKR 136123438 Ki = 794328.23 nM T16347 C49POR 136216675 IC50 = 24200 nM T16347 CJA8P0 136216676 IC50 = 30600 nM T16347 CTX10A 136216677 IC50 = 26900 nM T16347 C50MCG 136216678 IC50 = 6200 nM T16347 CY73XR 136216679 IC50 = 20600 nM T16347 CP3QE4 136216680 IC50 = 41300 nM T16347 C96JZW 136216681 IC50 = 23400 nM T16347 CEWV20 136216682 IC50 = 46000 nM T16347 CHD0M4 136216683 IC50 = 9100 nM T16347 C25EAK 136216684 IC50 = 9000 nM T16347 CUQ4C9 136216685 IC50 = 11600 nM T16347 CL7N1J 136216686 IC50 = 12400 nM T16347 CY5N1D 136216687 IC50 = 28400 nM T16347 CEG3F1 136224177 IC50 = 10300 nM T16347 CQ7L2H 136254273 IC50 > 100000 nM T16347 C5C1XF 136254274 IC50 > 100000 nM T16347 CL4A5E 136254275 IC50 > 100000 nM T16347 CH7N3Z 136254276 IC50 > 100000 nM T16347 CL4ZM7 136254277 IC50 > 100000 nM T16347 CAHC90 136254278 IC50 > 100000 nM T16347 CQ84LN 136254279 IC50 > 100000 nM T16347 CBEU97 136254280 IC50 > 100000 nM T16347 C3LK1C 136254281 IC50 = 83700 nM T16347 C5QIK7 137174949 IC50 > 120000 nM T16347 C6U0WH 137631389 IC50 = 10350 nM T16347 CN9HV1 137631809 Ki = 29260 nM T16347 CH6VY3 137632014 IC50 = 6040 nM T16347 CND2J9 137632455 IC50 = 11800 nM T16347 C9O8DG 137632552 IC50 = 240 nM T16347 CJL61E 137632606 IC50 = 1100 nM T16347 C8HJ5U 137632766 Ki = 1490 nM T16347 CPD4V1 137633197 IC50 = 160 nM T16347 CEY2O8 137633603 IC50 = 12340 nM T16347 CUA3W0 137633811 IC50 = 23590 nM T16347 CD51NF 137634169 IC50 = 4530 nM T16347 CQ2ZB6 137634422 IC50 > 100000 nM T16347 CU20HC 137634668 IC50 = 3000 nM T16347 C5D0FB 137634825 IC50 = 5100 nM T16347 C71KST 137634902 IC50 = 8450 nM T16347 CDZN68 137635090 IC50 = 4720 nM T16347 C03JHQ 137635891 IC50 = 6190 nM T16347 CVM4N6 137636541 Ki = 4380 nM T16347 CM6B9U 137636647 IC50 = 2600 nM T16347 CB8Y6H 137636689 IC50 = 13210 nM T16347 CZ6OK8 137636921 IC50 = 12460 nM T16347 CXQA50 137636968 IC50 = 6670 nM T16347 CXF3K6 137637073 IC50 = 7290 nM T16347 CZ49GD 137637199 IC50 = 10040 nM T16347 C5PJH8 137637756 Ki = 1000 nM T16347 CH1LF3 137637878 IC50 = 840 nM T16347 C65RSY 137637898 IC50 = 1500 nM T16347 CA0G1S 137638114 IC50 = 720 nM T16347 CO04IU 137638197 IC50 = 14530 nM T16347 C31SAR 137638729 IC50 = 8200 nM T16347 CQCI50 137638732 IC50 = 120000 nM T16347 CQ7NL9 137638893 Ki = 390 nM T16347 CQI1E5 137639232 IC50 = 850 nM T16347 CS7Z8A 137639334 Ki = 4400 nM T16347 CDE4W8 137639505 IC50 = 5700 nM T16347 CUC16I 137640493 IC50 > 20000 nM T16347 C1PMZ7 137640975 IC50 = 910 nM T16347 CSR64Z 137641155 IC50 = 3410 nM T16347 C0KJ6R 137641658 Ki = 2300 nM T16347 CSTD41 137641975 IC50 = 5430 nM T16347 CDH34Y 137642032 IC50 = 790 nM T16347 CIO61R 137642206 IC50 = 55100 nM T16347 CX4M7N 137642274 IC50 = 5830 nM T16347 C28DUQ 137642390 IC50 = 31230 nM T16347 CZ3K4A 137642893 IC50 = 750 nM T16347 C3QCG4 137643119 IC50 = 16520 nM T16347 CBU6I2 137643274 IC50 = 9200 nM T16347 C50SBG 137643363 IC50 = 1800 nM T16347 CZO03R 137643381 IC50 = 8000 nM T16347 C9OXT6 137643787 Ki = 1750 nM T16347 C2R7XB 137644229 IC50 = 7070 nM T16347 CRYZ81 137644333 IC50 = 820 nM T16347 C7D4SW 137644380 IC50 = 400 nM T16347 CFYQ61 137644492 IC50 = 12280 nM T16347 C8P4BL 137644511 IC50 = 37300 nM T16347 C16NUI 137644773 IC50 = 22250 nM T16347 CAW8Z9 137645547 IC50 = 6480 nM T16347 CE59LU 137645973 IC50 = 24290 nM T16347 CK37DU 137646355 IC50 > 20000 nM T16347 C48YBW 137646377 IC50 = 3890 nM T16347 C3F6CN 137646670 IC50 = 1900 nM T16347 C6TB1C 137646844 IC50 = 2200 nM T16347 CAF9N0 137647826 IC50 = 5250 nM T16347 CRD7Y5 137648180 IC50 = 6800 nM T16347 CR3ED8 137648245 IC50 = 29200 nM T16347 C38XYD 137648281 Ki = 1400 nM T16347 C2TU4K 137648375 IC50 = 3400 nM T16347 CHZ83R 137648907 IC50 = 1300 nM T16347 C2C7SD 137649366 IC50 = 7980 nM T16347 CRC71H 137649426 IC50 = 860 nM T16347 CG0Z1I 137649766 Ki = 5900 nM T16347 CY5U6F 137650241 IC50 = 18400 nM T16347 C8LAH5 137650349 IC50 = 200 nM T16347 C6LZ4J 137650470 IC50 = 750 nM T16347 CN1X0J 137651804 IC50 = 350 nM T16347 CMP5G0 137652244 IC50 = 20560 nM T16347 CFV26J 137652273 IC50 = 4270 nM T16347 CLH9Z3 137652709 IC50 = 5610 nM T16347 C3DZ9S 137652811 IC50 = 4650 nM T16347 CM3EQ1 137652959 IC50 = 5000 nM T16347 CXQ40F 137653094 IC50 = 140 nM T16347 CGW41H 137653135 IC50 = 870 nM T16347 CQ7T4S 137653723 IC50 = 1200 nM T16347 CK4IY9 137654311 IC50 = 11290 nM T16347 CFAX47 137654492 IC50 > 20000 nM T16347 CH0L4W 137654779 IC50 = 1110 nM T16347 CRT40L 137654807 Ki = 300 nM T16347 CGSL14 137654967 IC50 = 8700 nM T16347 C2N3GP 137655294 IC50 = 1100 nM T16347 C2QO8A 137655901 IC50 = 14790 nM T16347 C63NUF 137656713 IC50 = 16320 nM T16347 CAW80L 137656933 IC50 = 1300 nM T16347 CL4Z1R 137657281 IC50 = 190 nM T16347 C4PJL8 137657720 IC50 = 3000 nM T16347 C72KQM 137660406 IC50 = 11220 nM T16347 CCXY75 137660653 IC50 = 1400 nM T16347 C4CY9T 137661102 IC50 = 190 nM T16347 C1A2CR 137661401 IC50 = 5340 nM T16347 C2XLT6 137661766 IC50 = 7100 nM T16347 CDUW41 137661805 Ki = 1500 nM T16347 CFP95B 137661822 IC50 = 6370 nM T16347 CO1LB8 137662103 IC50 = 3500 nM T16347 CY23BH 137662149 IC50 = 1300 nM T16347 CA5ME9 139051002 IC50 = 19880 nM T16347 C0WMZ4 139593950 IC50 = 190 nM T16347 C6H1UW 141746816 IC50 = 9400 nM T16347 C1FT7V 141746817 IC50 = 16300 nM T16347 CME89I 141746818 IC50 = 7200 nM T16347 C6VFT4 141746819 IC50 = 5900 nM T16347 CL15BV 141746820 IC50 = 3900 nM T16347 C21JSO 141746823 IC50 = 10900 nM T16347 CJ5IW8 141746824 IC50 = 5400 nM T16347 C5R9AU 141746825 IC50 = 6300 nM T16347 C36HJM 141746826 IC50 = 32800 nM T16347 C8X4BN 141746828 IC50 = 5800 nM T16347 C8GXK3 141746830 IC50 = 6500 nM T16347 CM3ZF9 141746831 IC50 = 6900 nM T16347 C2NZI9 141746832 IC50 = 8200 nM T16347 CLN7E5 141746833 IC50 = 4700 nM T16347 CNMV29 141746834 IC50 = 5900 nM T16347 CHPG81 141746836 IC50 = 4600 nM T16347 C2OG8K 141746837 IC50 = 7400 nM T16347 C06SDN 141746838 IC50 = 5400 nM T16347 CM6F8C 141746840 IC50 = 9500 nM T16347 C28LVZ 141746842 IC50 = 6900 nM T16347 CFZA47 141746843 IC50 = 570 nM T16347 CSQ7K8 141746844 IC50 = 5300 nM T16347 C3ZW6K 141746845 IC50 = 3900 nM T16347 C26ESX 141746846 IC50 = 6900 nM T16347 CEQO31 141746847 IC50 = 24800 nM T16347 CH53WF 141746848 IC50 = 12300 nM T16347 CPT63G 141746851 IC50 = 14600 nM T16347 C6NQ9I 145720956 IC50 = 14000 nM T16347 CJT93U 145721022 IC50 = 13000 nM T16347 CECA72 145721223 IC50 = 27000 nM T16347 C8VDR6 145721225 IC50 = 23000 nM T16347 CP73QC 145949173 IC50 = 15490 nM T16347 CJR71S 145949439 IC50 = 20030 nM T16347 C09HAX 145949577 IC50 = 3600 nM T16347 CFOP95 145949822 IC50 = 4300 nM T16347 C7RE6D 145950050 IC50 = 10470 nM T16347 CS5H2Y 145950066 IC50 = 169.2 nM T16347 C0LJD8 145950440 IC50 = 7790 nM T16347 C42OXT 145950507 IC50 = 8090 nM T16347 C4DWG8 145950748 IC50 = 68.2 nM T16347 CK8D3M 145950815 IC50 = 487 nM T16347 CU9BM7 145951467 IC50 = 4800 nM T16347 CUI29N 145951937 IC50 = 31630 nM T16347 CCRF92 145952989 IC50 = 16980 nM T16347 CL32PZ 145953390 IC50 = 8000 nM T16347 CS9ID4 145953582 IC50 = 6250 nM T16347 CN0M2W 145953858 IC50 = 10960 nM T16347 CEZ8L7 145953861 IC50 = 6020 nM T16347 CJS5Y4 145954007 IC50 = 7600 nM T16347 C4NJU2 145954341 IC50 = 15000 nM T16347 CL5S1B 145955081 IC50 = 7600 nM T16347 CN8TM7 145955117 IC50 = 21380 nM T16347 C3QP2X 145955503 IC50 = 7400 nM T16347 CK04YT 145955715 IC50 = 4870 nM T16347 CSVD04 145955743 IC50 = 42000 nM T16347 CNSP90 145955796 IC50 = 10160 nM T16347 CUMF50 145956030 IC50 = 2630 nM T16347 CN6K5Q 145956149 IC50 = 20820 nM T16347 C1SU7K 145956845 IC50 = 9330 nM T16347 CO3Q4M 145957138 IC50 = 47350 nM T16347 C1USV5 145957197 IC50 = 35580 nM T16347 CTOK38 145957219 IC50 = 710.9 nM T16347 C20OTG 145957700 IC50 = 11080 nM T16347 C8ZP9F 145957853 IC50 = 115340 nM T16347 C65YFU 145957867 IC50 = 19140 nM T16347 C2N1QH 145958444 IC50 = 7600 nM T16347 CB84OL 145958621 IC50 = 7940 nM T16347 C8W5NV 145958623 IC50 = 12000 nM T16347 CT8CM4 145958683 IC50 = 9400 nM T16347 C4RZ6D 145958850 IC50 = 807 nM T16347 C8TE4C 145958942 IC50 = 49450 nM T16347 CPC4Q7 145959149 IC50 = 14360 nM T16347 CAVH30 145959629 IC50 = 3890 nM T16347 CVJ80O 145960007 IC50 = 6920 nM T16347 CBA7F3 145960113 IC50 = 12440 nM T16347 CIZE64 145960181 IC50 = 209.1 nM T16347 CF8GB1 145960243 IC50 = 4740 nM T16347 CRV8M9 145960352 IC50 = 11000 nM T16347 CT6I5O 145961409 IC50 = 18.6 nM T16347 CSB21A 145961412 IC50 = 981 nM T16347 CG4OJ7 145963136 IC50 = 22750 nM T16347 CX5EF2 145963522 IC50 = 165.9 nM T16347 CGW13B 145964794 IC50 = 29000 nM T16347 CZ2IU0 145964831 IC50 > 100000 nM T16347 CC6B7J 145965718 IC50 = 61000 nM T16347 CO7AV3 145965953 IC50 = 213000 nM T16347 CA8SZ5 145966877 IC50 > 100000 nM T16347 C2J0KF 145966924 Ki = 2100 nM T16347 C9ICD0 145966982 IC50 = 48260 nM T16347 CX93IC 145967464 IC50 > 100000 nM T16347 CT9D5V 145969613 IC50 = 23800 nM T16347 CUO63K 145969860 Ki = 32700 nM T16347 C58OBV 145971193 IC50 = 66.2 nM T16347 CUE85W 145971302 IC50 = 50230 nM T16347 CFE82Y 145971670 IC50 = 24700 nM T16347 C6DNT5 145972085 IC50 = 43600 nM T16347 C73LAX 145972390 IC50 = 42150 nM T16347 CV3FS9 145972458 IC50 = 184.1 nM T16347 C4SDK2 145972554 IC50 = 313000 nM T16347 COH0T4 145972708 IC50 = 7440 nM T16347 CI6D1R 145972906 IC50 = 44380 nM T16347 CHNX81 145973061 IC50 = 46300 nM T16347 CVM64I 145973093 IC50 = 127000 nM T16347 CLB36X 145973142 IC50 = 56000 nM T16347 C5QY9L 145973266 IC50 = 58200 nM T16347 CB1KG6 145974093 IC50 = 13000 nM T16347 C1XSU8 145974786 IC50 = 21370 nM T16347 CZ2J7L 145975310 IC50 = 38100 nM T16347 CR54JZ 145975482 Ki = 3400 nM T16347 C73QYE 145975658 IC50 = 19300 nM T16347 C26IVS 145975708 IC50 = 48000 nM T16347 CY6KU9 145975895 IC50 > 100000 nM T16347 CP28YI 145976403 IC50 = 48100 nM T16347 C82EIW 145976484 IC50 = 38220 nM T16347 C2OZ8G 145976572 IC50 = 33560 nM T16347 C7SM3Z 145977996 Ki = 8900 nM T16347 C09TSQ 145978898 IC50 = 700 nM T16347 C2J1LR 145982026 IC50 = 38200 nM T16347 C0ZW2J 145982366 IC50 > 50000 nM T16347 CT8Y1X 145988950 IC50 = 17000 nM T16347 CZGK60 145992331 IC50 = 9400 nM T16347 C2TCV7 154720649 IC50 = 24320 nM T16347 CI46NM 155510388 IC50 = 1070 nM T16347 CO7SN0 155510754 IC50 = 720 nM T16347 CB6S1P 155511027 IC50 = 16300 nM T16347 CG4X0L 155511054 IC50 = 43600 nM T16347 C1Y0RZ 155511084 IC50 = 76000 nM T16347 CBTK25 155511429 IC50 = 7120 nM T16347 CQ8X4N 155511553 IC50 = 1670 nM T16347 CE38YK 155511993 IC50 = 1070 nM T16347 CJ3K7C 155512263 IC50 = 420 nM T16347 C9AI6C 155512404 IC50 = 14000 nM T16347 C5TBN2 155512577 IC50 = 3000 nM T16347 C82YVE 155513052 IC50 = 1540 nM T16347 CQ3LP9 155513935 IC50 = 11800 nM T16347 CZ8T7U 155514185 IC50 = 4000 nM T16347 C24KSX 155514321 IC50 = 88000 nM T16347 CHWJ95 155514409 IC50 = 6650 nM T16347 CZ09KH 155514693 IC50 = 9130 nM T16347 C7VH6E 155515065 IC50 = 16000 nM T16347 CP9B8J 155515271 IC50 = 5490 nM T16347 CL6I0W 155515906 IC50 = 1510 nM T16347 CT1I8A 155516446 IC50 = 10260 nM T16347 CU8Z5H 155516617 IC50 > 100000 nM T16347 CB2I5V 155517051 IC50 = 2800 nM T16347 C8P4JG 155517713 IC50 = 6680 nM T16347 C3PVL6 155517759 IC50 = 6840 nM T16347 CGUP05 155517773 IC50 = 450 nM T16347 CH3V5O 155517781 IC50 = 2700 nM T16347 CQT5W0 155517916 IC50 = 9200 nM T16347 CP31JD 155518035 IC50 = 820 nM T16347 C7L3BR 155518108 IC50 = 1080 nM T16347 CI1A8S 155518216 IC50 = 4900 nM T16347 CH5BD8 155518698 IC50 = 59000 nM T16347 C9XLV1 155518835 IC50 = 7440 nM T16347 C40OYE 155519056 IC50 = 6400 nM T16347 CDYT42 155519082 IC50 = 250 nM T16347 C1HL4K 155519234 IC50 = 2800 nM T16347 C2LEI3 155519273 IC50 = 22800 nM T16347 C58GUT 155519433 IC50 = 36000 nM T16347 CVI14S 155519450 IC50 = 12400 nM T16347 C2Y5JT 155519607 IC50 = 78000 nM T16347 CEOK93 155519659 IC50 = 51000 nM T16347 CUT96N 155520005 IC50 = 3500 nM T16347 CDA80Z 155520686 IC50 = 14000 nM T16347 CXW03M 155520805 IC50 = 1370 nM T16347 C8ZV6K 155520858 IC50 = 38000 nM T16347 CS0FB9 155521020 IC50 = 13000 nM T16347 CZ75SL 155521073 IC50 = 540 nM T16347 C5AD6C 155521134 IC50 = 46000 nM T16347 C8XB0K 155521306 IC50 = 86000 nM T16347 CX6NP9 155522115 IC50 > 50000 nM T16347 CA7K3L 155522245 IC50 = 1390 nM T16347 CPA2Q1 155522760 IC50 = 3510 nM T16347 C2WP6O 155522824 IC50 = 2800 nM T16347 CX4HE9 155522866 IC50 = 6500 nM T16347 CW1V5X 155522892 IC50 = 2800 nM T16347 C97FCS 155523863 IC50 = 57000 nM T16347 C6T4LN 155523864 IC50 = 42420 nM T16347 CS1MY2 155524015 IC50 = 37000 nM T16347 C6O7IF 155524023 IC50 = 22800 nM T16347 CXJ3G8 155524072 IC50 = 5000 nM T16347 CV9T1G 155524326 IC50 = 11000 nM T16347 C8CK4L 155524588 IC50 > 50000 nM T16347 CF3W1J 155525280 IC50 = 151000 nM T16347 C1DBI9 155525852 IC50 = 380 nM T16347 CZ39RU 155525942 IC50 = 47000 nM T16347 CC0BW9 155526176 IC50 = 37000 nM T16347 C9KP7O 155526482 IC50 > 100000 nM T16347 C6HQX8 155526489 IC50 = 70000 nM T16347 C4BVF8 155526535 Ki = 12000 nM T16347 CRXH61 155526717 IC50 > 100000 nM T16347 CV9B1Q 155527194 IC50 = 430 nM T16347 C8FXO7 155527541 IC50 = 5930 nM T16347 C23XTW 155527930 IC50 = 10990 nM T16347 C6TJ8W 155528254 IC50 > 50000 nM T16347 CR3T0B 155528310 IC50 = 18550 nM T16347 CEM5A4 155528339 IC50 = 1170 nM T16347 CNA15X 155528422 IC50 = 6600 nM T16347 C29HIT 155528492 IC50 = 44000 nM T16347 C1T5EO 155528736 IC50 = 5520 nM T16347 C6OSW5 155528751 IC50 = 53000 nM T16347 C0C8RL 155528754 IC50 = 2790 nM T16347 CA5QP6 155528768 IC50 = 40000 nM T16347 C4UM7L 155528968 IC50 = 1260 nM T16347 C8P2FO 155529472 IC50 = 2440 nM T16347 C6A0JM 155529655 IC50 = 13000 nM T16347 CRP05Z 155530032 IC50 = 76000 nM T16347 CX93AN 155530064 IC50 = 5000 nM T16347 C9TW3U 155530403 IC50 = 2600 nM T16347 CKVG10 155530868 IC50 = 92000 nM T16347 CKD9O4 155530916 IC50 = 59000 nM T16347 C2HWB8 155531242 IC50 = 460 nM T16347 CTB6J8 155531587 IC50 = 770 nM T16347 C9KB8S 155531981 IC50 = 10350 nM T16347 C9MOL6 155532600 IC50 = 8400 nM T16347 C38HEA 155532611 IC50 = 300 nM T16347 C17KUO 155532644 IC50 = 7490 nM T16347 CXJ0Q8 155533186 IC50 = 16660 nM T16347 CG76KF 155533254 IC50 = 3340 nM T16347 C4RBN5 155533387 IC50 = 3600 nM T16347 C6Q4GW 155533586 IC50 = 4700 nM T16347 CT01ZQ 155533593 IC50 = 33000 nM T16347 CW25RG 155534915 IC50 = 44000 nM T16347 CCS74T 155534973 IC50 = 440 nM T16347 CK3GW1 155535090 IC50 = 9340 nM T16347 C94HBY 155535475 IC50 = 11380 nM T16347 CL12VT 155535839 IC50 = 3810 nM T16347 C7Y5JF 155535845 IC50 = 18900 nM T16347 CWIG06 155536052 IC50 = 32240 nM T16347 CA1K8G 155536107 IC50 > 80000 nM T16347 CG3W2A 155536205 IC50 = 3380 nM T16347 CCSW05 155536292 IC50 = 6870 nM T16347 CE37VK 155536544 IC50 = 25600 nM T16347 CGTE62 155536611 IC50 = 285 nM T16347 CLZ31N 155536741 IC50 = 120 nM T16347 C6I8VT 155537121 IC50 = 800 nM T16347 CKV5E7 155537236 IC50 = 6200 nM T16347 CQ63GA 155537698 Ki = 70 nM T16347 CRU6F2 155538623 IC50 = 640 nM T16347 C3Y6ZF 155538861 IC50 = 870 nM T16347 C35XOI 155538992 IC50 = 37000 nM T16347 CKZ2Q8 155539050 IC50 = 8800 nM T16347 C0BPO1 155539639 IC50 = 1530 nM T16347 CO0R1M 155539881 IC50 = 4790 nM T16347 CJG35L 155540073 IC50 = 7420 nM T16347 C6C7ZQ 155540504 Ki = 7600 nM T16347 C0YK4X 155540612 IC50 = 24000 nM T16347 C5BP9T 155541433 IC50 = 6310 nM T16347 CP4R6C 155541505 Ki = 2570 nM T16347 CS7N6V 155541568 IC50 = 6900 nM T16347 CZUP50 155542230 IC50 = 9400 nM T16347 C2ZX5U 155542716 IC50 = 83000 nM T16347 C59FAJ 155542764 IC50 = 19000 nM T16347 CK8H7F 155542996 IC50 = 12000 nM T16347 C2L3EB 155543224 IC50 = 1930 nM T16347 CU1M7O 155543297 IC50 = 10000 nM T16347 CQ68VS 155543531 IC50 = 40000 nM T16347 CUJ1D3 155543880 IC50 = 0.42 nM T16347 CEJZ14 155543962 IC50 = 22200 nM T16347 COFL10 155544758 IC50 = 71000 nM T16347 CD12KN 155544808 IC50 = 63000 nM T16347 C1N8IW 155544848 IC50 > 100000 nM T16347 CBW7U9 155544853 IC50 = 35000 nM T16347 CLF25Z 155545436 IC50 = 230 nM T16347 CL78UG 155545756 IC50 = 2800 nM T16347 C4U0NO 155545913 IC50 = 3750 nM T16347 CT3E0D 155546030 IC50 = 11000 nM T16347 C67VHZ 155546266 IC50 = 11000 nM T16347 CKXI09 155546310 IC50 = 7900 nM T16347 CKU40H 155546574 IC50 = 4270 nM T16347 C24LXU 155546956 IC50 = 37000 nM T16347 C8PB0Y 155547153 IC50 = 7200 nM T16347 C1N3DJ 155547316 IC50 = 73000 nM T16347 CPA43X 155547531 IC50 = 720 nM T16347 CDZ23J 155547591 IC50 = 610 nM T16347 C1XM3W 155547918 IC50 = 1260000 nM T16347 CARH78 155548168 IC50 = 16800 nM T16347 COZE38 155548201 IC50 = 4360 nM T16347 C1N8YP 155548589 IC50 = 2520 nM T16347 CRH8J5 155548680 IC50 = 1030 nM T16347 C9ZBY7 155548951 IC50 = 27000 nM T16347 C2BQU0 155549283 IC50 = 6900 nM T16347 C1HRL5 155549365 IC50 = 12600 nM T16347 CO1QI3 155549402 IC50 = 2450 nM T16347 C4YEZ7 155549652 IC50 > 80000 nM T16347 C04LDI 155550280 IC50 = 18470 nM T16347 C50TQN 155550512 Ki = 140 nM T16347 CB8J9Q 155550870 IC50 = 35000 nM T16347 CB1J7W 155550987 IC50 = 6900 nM T16347 C0KRS3 155551320 IC50 = 5 nM T16347 C98WJA 155551471 IC50 = 55000 nM T16347 CA7J4V 155552115 IC50 > 100000 nM T16347 CLK6H2 155552277 IC50 > 80000 nM T16347 CL6GJ5 155552588 IC50 > 50000 nM T16347 CG4T9K 155552640 IC50 = 3330 nM T16347 CR0W1D 155552684 IC50 = 8230 nM T16347 CML3E0 155553010 IC50 = 1700 nM T16347 CO7M4Q 155553141 IC50 = 12000 nM T16347 CUX36E 155553266 IC50 = 3180 nM T16347 CZS4E8 155553560 IC50 = 2950 nM T16347 C6MQD2 155553640 IC50 = 8600 nM T16347 CV9Y7C 155553768 IC50 = 1220 nM T16347 C9ZG1S 155554310 IC50 = 7900 nM T16347 CJC6B3 155555083 IC50 > 50000 nM T16347 C58FEN 155555616 IC50 = 10700 nM T16347 CKH13G 155555860 IC50 = 22990 nM T16347 CN6G0X 155556117 IC50 = 27400 nM T16347 CA75HC 155556730 IC50 = 830 nM T16347 C3WY9T 155557150 IC50 = 3360 nM T16347 C6T4YC 155557626 IC50 = 42000 nM T16347 CMEK61 155557904 IC50 = 54000 nM T16347 C0B5QW 155558168 IC50 = 19100 nM T16347 C8ORY6 155558805 IC50 = 10000 nM T16347 C7GDN0 155558939 IC50 = 11900 nM T16347 C8FUW1 155558944 IC50 = 28000 nM T16347 CY1PA9 155559338 IC50 = 1450 nM T16347 C42KAN 155559479 IC50 = 29000 nM T16347 CG2E1P 155560132 IC50 = 62000 nM T16347 C2EAN8 155560211 IC50 = 2290 nM T16347 CLHC31 155560435 IC50 = 21000 nM T16347 C3VS9F 155560547 IC50 = 11000 nM T16347 C5E0GW 155560770 Ki = 32 nM T16347 C8YPK2 155561887 Ki = 4130 nM T16347 C1XKG0 155562197 IC50 = 5030 nM T16347 CDW65X 155562259 IC50 = 44000 nM T16347 C8V9CR 155562599 IC50 = 5760 nM T16347 C2LSK5 155562777 IC50 = 76000 nM T16347 CR58CV 155563028 IC50 > 50000 nM T16347 CZY09O 155563068 IC50 = 52000 nM T16347 C0GEV5 155563686 IC50 = 45000 nM T16347 C08UCW 155563714 IC50 = 40000 nM T16347 CE74XH 155564341 IC50 = 1180 nM T16347 C8BG3P 155564911 IC50 = 14000 nM T16347 CCO51A 155565389 IC50 = 1450 nM T16347 CL1S9J 155565716 IC50 = 1990 nM T16347 C2RTX8 155565846 IC50 = 700 nM T16347 C51DXF 155566190 IC50 = 11300 nM T16347 CQO8G5 155566227 IC50 = 11000 nM T16347 C1E9RX 155566282 IC50 = 7810 nM T16347 CL17NY 155566313 IC50 = 35000 nM T16347 C7W5HT 155566457 IC50 = 2140 nM T16347 C7I0XS 155566497 IC50 = 360 nM T16347 CRHU69 155566574 IC50 > 80000 nM T16347 CAN4F0 155567088 IC50 = 6280 nM T16347 C0RVL8 155567421 IC50 = 3550 nM T16347 C1V6GI 155567809 IC50 = 5400 nM T16347 CEN0C6 155568015 IC50 > 80000 nM T16347 CE13QZ 155568166 IC50 = 2380 nM T16347 C0E7BX 155568773 IC50 = 28000 nM T16347 CF3OQ9 155568971 IC50 = 5770 nM T16347 CKI57Q 155569114 IC50 = 1200 nM T16347 CU47ID 10122761 Ki = 398.11 nM T16347 CNR70V 22271897 Ki = 1000 nM T16347 C8AYE4 22271914 Ki = 63.1 nM T16347 CTM43U 22271953 Ki = 158.49 nM T16347 C34EPH 22271970 Ki = 630.96 nM T16347 C4CDY5 24850295 IC50 = 15000 nM T16347 C9M5FS 45266937 Ki = 3981.07 nM T16347 CI72DE 45266938 Ki = 1258.93 nM T16347 CIGW92 45266942 Ki = 1995.26 nM T16347 CAO17S 45267004 Ki = 199.53 nM T16347 CZ84IJ 45267800 Ki = 398.11 nM T16347 C0CEA1 45268680 Ki = 1995.26 nM T16347 CXR7H9 45268795 Ki = 10000 nM T16347 C32XSL 45269558 Ki = 316.23 nM T16347 CE5LF1 45269640 Ki = 3981.07 nM T16347 CW7U6I 45270475 Ki = 1258.93 nM T16347 CHGW15 45272099 Ki = 19952.62 nM T16347 C86ZUY 45272105 Ki = 19.95 nM T16347 CH6F4K 45272192 Ki = 398.11 nM T16347 C6CUJ8 45273052 Ki = 3981.07 nM T16347 D00DDO 268734 IC50 = 351000 nM T16347 D00KZO 21147013 IC50 = 7300 nM T16347 D00MNE 7330513 IC50 = 16000 nM T16347 D00RZN 442457 IC50 = 17300 nM T16347 D00VNC 44411858 IC50 = 5200 nM T16347 D01BZE 73659 IC50 = 5930 nM T16347 D01EJH 11500744 IC50 = 7600 nM T16347 D01NUT 5467256 IC50 = 4300 nM T16347 D01SLG 446512 IC50 = 1.24 nM T16347 D01VNN 360384 IC50 = 242000 nM T16347 D02HCQ 1794427 IC50 = 11100 nM T16347 D02KKU 12313704 IC50 = 5320 nM T16347 D02SGJ 19009 IC50 = 234000 nM T16347 D03BHQ 45273571 Ki = 4300 nM T16347 D03EGZ 442531 IC50 = 3500 nM T16347 D03KGX 12315077 IC50 = 10900 nM T16347 D03KJL 10107739 IC50 = 130000 nM T16347 D03ZIH 52946645 Ki = 18 nM T16347 D04BYU 8546 IC50 = 310000 nM T16347 D04TGN 181620 IC50 > 1000000 nM T16347 D04TTB 44411959 IC50 = 11700 nM T16347 D05AOH 10333896 IC50 = 1140000 nM T16347 D05DOM 6227 Ki = 77000000 nM T16347 D05IWY 5464078 Ki = 2700 nM T16347 D05SEV 2259222 IC50 = 8600 nM T16347 D05TNT 738951 IC50 = 5700 nM T16347 D06AWX 5326018 IC50 = 3770 nM T16347 D06BFB 44411962 IC50 = 12800 nM T16347 D06LNL 101840 IC50 = 2650000 nM T16347 D06NGA 4369452 IC50 = 2500 nM T16347 D06PRC 5281650 Ki = 3200 nM T16347 D06ZRX 5281717 IC50 = 27130 nM T16347 D07DJS 5280459 IC50 = 17.49 ug.mL-1 T16347 D07DNK 1628 Ki = 10000 nM T16347 D07LUJ 64945 IC50 = 2300 nM T16347 D07WQA 4437 IC50 > 4000000 nM T16347 D08ABU 12193680 IC50 = 15600 nM T16347 D08BSQ 54678922 IC50 = 4.5 nM T16347 D08GDJ 9547915 Ki = 180 nM T16347 D08GEN 5318998 IC50 = 19100 nM T16347 D08GWQ 44409669 IC50 = 13660 nM T16347 D08SAG 25033124 Ki = 1500 nM T16347 D08UOX 5281148 IC50 = 8.22 ug.mL-1 T16347 D08VRV 45485203 IC50 = 13800 nM T16347 D09CAI 440646 IC50 = 0.67 nM T16347 D09GPV 21594148 IC50 = 18800 nM T16347 D09HAX 73205 IC50 = 19400 nM T16347 D09OWE 92802 IC50 = 15600 nM T16347 D09TUB 11099375 IC50 = 970 nM T16347 D09VQM 442428 IC50 = 91800 nM T16347 D09VYW 9847548 IC50 = 8040 nM T16347 D09WED 45485202 IC50 = 8200 nM T16347 D09YKH 42607959 IC50 = 18900 nM T16347 D0A1QK 44139929 IC50 = 51.63 nM T16347 D0A4ML 10854796 IC50 = 741.31 nM T16347 D0A8WJ 184877 IC50 = 16900 nM T16347 D0A9CZ 119268 IC50 > 30000 nM T16347 D0C0DM 11455599 IC50 = 2420 nM T16347 D0D4SI 44568920 IC50 = 12800 nM T16347 D0DU3J 44424649 IC50 = 19200 nM T16347 D0E0BU 444763 Ki = 7943.28 nM T16347 D0E1UG 44411982 IC50 = 16000 nM T16347 D0E1ZS 5281297 IC50 = 9200 nM T16347 D0F3QP 5889042 IC50 = 74100 nM T16347 D0F9RO 6918774 IC50 = 5490 nM T16347 D0G4GB 10757 Ki = 480000 nM T16347 D0G7HN 3718733 IC50 = 200000 nM T16347 D0H1WV 45273151 IC50 = 2700 nM T16347 D0H3NS 10752 IC50 > 1000000 nM T16347 D0J5KG 44411771 IC50 = 14200 nM T16347 D0J5VK 67145 IC50 = 3600000 nM T16347 D0JB4G 67220 IC50 = 9700 nM T16347 D0JL8I 46879996 IC50 = 19300 nM T16347 D0K0PR 10600994 IC50 = 8100 nM T16347 D0K3TS 73204 IC50 = 14400 nM T16347 D0K4PY 114829 IC50 > 60000 nM T16347 D0L3IQ 442153 IC50 = 22600 nM T16347 D0LC7K 119034 IC50 > 20000 nM T16347 D0LS2U 17413 IC50 > 1000000 nM T16347 D0M0XS 44411975 IC50 = 8500 nM T16347 D0M7ZZ 637080 IC50 = 8800 nM T16347 D0MG9O 54689623 IC50 = 3000 nM T16347 D0N4XG 417214 IC50 = 400 nM T16347 D0N7XM 24992964 IC50 > 30000 nM T16347 D0N7YT 44409922 IC50 = 19590 nM T16347 D0N8OO 164215 IC50 = 14200 nM T16347 D0O1BJ 445434 IC50 = 1.17 nM T16347 D0O7ZE 5311365 IC50 = 0.3 nM T16347 D0O7ZL 15560128 IC50 = 4930 nM T16347 D0OJ1V 44411588 IC50 = 7100 nM T16347 D0OY2V 46880035 IC50 = 19500 nM T16347 D0P5MJ 10410005 IC50 = 20800 nM T16347 D0P9SW 46880036 IC50 = 6400 nM T16347 D0Q2YJ 6763 IC50 > 30000 nM T16347 D0Q3KF 9841650 IC50 = 1190 nM T16347 D0Q5PQ 15840592 IC50 = 7800 nM T16347 D0Q8AT 25564831 IC50 = 14330 nM T16347 D0QQ7A 11995582 IC50 = 14800 nM T16347 D0RA6H 259846 IC50 = 3680 nM T16347 D0S9GU 16737250 IC50 = 15700 nM T16347 D0SJ2Q 10494 IC50 = 0.85 ug.mL-1 T16347 D0U2WU 3549290 IC50 = 890000 nM T16347 D0U6AI 25262526 IC50 = 19000 nM T16347 D0U8IF 10114 IC50 = 45800 nM T16347 D0V0LU 11740841 IC50 = 7600 nM T16347 D0V9EN 689043 IC50 = 3060 nM T16347 D0VA9F 157143 IC50 = 4900 nM T16347 D0W1OR 7424 IC50 > 100000 nM T16347 D0W9VA 10667 IC50 = 1640 nM T16347 D0Y1RO 1829 Ki = 14000 nM T16347 D0Y5SB 444764 Ki = 22908.68 nM T16347 D0Z1HV 382831 IC50 = 3900 nM T16347 D0ZE8C 25033201 IC50 = 3500 nM T16347 D0ZS7M 45268827 IC50 = 4200 nM T82773 D0E3TC 44259 IC50 = 3070 nM T82773 CLS29B 46872626 IC50 > 10000 nM T82773 CON8H1 59326984 IC50 = 6560 nM T82773 CIM7H1 66575095 IC50 = 200 nM T82773 CV63UL 67240318 IC50 > 10000 nM T82773 CI8EG4 70682610 IC50 = 14900 nM T82773 CJ1RE5 70682611 IC50 = 3830 nM T82773 C2MPQ3 70686838 IC50 = 1510 nM T82773 CCJH52 70691010 IC50 = 4890 nM T82773 C39DER 70691011 IC50 = 2340 nM T82773 CLZ4Q1 70691012 IC50 = 13000 nM T82773 CAJF37 70693140 IC50 = 1170 nM T82773 C2U7ES 70693141 IC50 = 4540 nM T82773 CQ75AH 70693142 IC50 = 700 nM T82773 CC48LS 70695212 IC50 = 1450 nM T82773 C56HSY 70695213 IC50 = 10100 nM T82773 CX61EW 70697244 IC50 = 9100 nM T82773 C7VA0I 71450358 IC50 = 26 nM T82773 CZ2OE6 71452173 IC50 = 8 nM T82773 CSPN93 71452174 IC50 = 50 nM T82773 CR53ZS 71452175 IC50 = 5 nM T82773 CM14JZ 71452176 IC50 = 4 nM T82773 CX1KZ0 71453985 IC50 = 17 nM T82773 CFGP02 71455731 IC50 = 80 nM T82773 CS27GC 71457514 IC50 = 8 nM T82773 C16OVY 71457515 IC50 = 853 nM T82773 C3KIM9 71461149 IC50 = 33 nM T82773 CW6MK4 71462888 IC50 = 24 nM T82773 C9V6KY 71462889 IC50 = 3 nM T82773 C2MD1Q 155513187 IC50 > 10000 nM T82773 D00ERW 44444843 Ki > 7166 nM T82773 D0H4VB 71461150 IC50 = 3 nM T47094 D06GDY 43815 IC50 = 900 nM T47094 D0GU4K 135413536 Ki = 0.07943 nM T47094 D02DLP 6918330 Ki = 0.02512 nM T47094 D05ZWG 108147 Ki > 10000 nM T47094 D06HCC 3086681 IC50 = 0.15 nM T47094 D0CB2B 23653789 IC50 = 0.06 nM T47094 D0DM6I 132961 IC50 = 13000 nM T47094 D0G3YC 6451149 Ki = 0.95 nM T47094 D0K5HI 5311424 Ki > 10000 nM T47094 D0LI1C 44469321 IC50 > 10000 nM T47094 D0P1YE 9852175 Ki = 0.0631 nM T47094 D0T0PN 9821217 IC50 = 0.14 nM T47094 D0V7US 9917079 IC50 = 0.07943 nM T47094 D00VPT 6604009 Ki > 100000 nM T47094 D00CQB 9805809 IC50 = 0.5495 nM T47094 D00ZGA 9917021 Ki = 0.1259 nM T47094 D02TKI 132846 IC50 = 0.87 nM T47094 D03SXN 104943 IC50 = 0.2 nM T47094 D04RCG 10327792 IC50 = 800 nM T47094 D04RUP 9851211 IC50 = 82400 nM T47094 D04VDY 135539114 IC50 = 0.05 nM T47094 D05WJQ 104974 IC50 = 593 nM T47094 D07PLK 158365 IC50 = 230 nM T47094 D08KXE 107686 IC50 = 30 nM T47094 D08ZBV 132837 Ki = 0.73 nM T47094 D09JXL 5311430 IC50 > 1000 nM T47094 D0A1KU 11683187 Ki = 6500 nM T47094 D0C9FF 9939040 Ki = 4.169 nM T47094 D0IP6X 219077 Ki = 209.6 nM T47094 D0J3QU 44351946 Ki = 1620 nM T47094 D0J5CX 9894349 IC50 = 0.45 nM T47094 D0N1PA 9869033 IC50 = 12 nM T47094 CGC70I 105083 Ki = 0.17 nM T47094 CI4WX2 127943 Ki = 0.03981 nM T47094 CA4NS3 127944 Ki = 0.05012 nM T47094 C20AYU 153996 Ki = 0.3 nM T47094 CLR5Z4 163732 Ki = 1.1 nM T47094 CBJ74I 163829 Ki = 0.14 nM T47094 CQT15N 178025 IC50 = 19.05 nM T47094 C2UQ3S 195814 EC50 = 0.6 nM T47094 CYOJ62 489662 IC50 = 1 nM T47094 CK24WR 490428 IC50 = 2.2 nM T47094 CZN6S9 743974 IC50 > 50118.72 nM T47094 CSE81V 1122655 IC50 = 250 nM T47094 C5N1KX 1760285 Ki > 100000 nM T47094 CMLC05 1760287 Ki > 100000 nM T47094 C59DHG 2755911 Ki = 5.2 nM T47094 C0UR7K 4529080 Ki > 100000 nM T47094 C5PO1F 6604014 Ki > 100000 nM T47094 CE57YD 6604858 Ki > 100000 nM T47094 CD6H5Z 6918331 Ki = 0.05012 nM T47094 C7Q5AJ 6995075 IC50 > 10000 nM T47094 C36VYU 7016092 IC50 > 10000 nM T47094 C2W6PI 8867347 Ki = 6700 nM T47094 C5K3NQ 9799676 IC50 = 4.4 nM T47094 C68UYJ 9801487 IC50 = 25.12 nM T47094 CQE1T4 9808347 Ki = 1.1 nM T47094 C29KSY 9808518 Ki = 0.58 nM T47094 COF63N 9809308 Ki = 3715.35 nM T47094 CL81MT 9809876 Ki = 0.17 nM T47094 CIGT19 9810434 Ki = 0.5 nM T47094 C35MSJ 9810544 Ki = 0.8 nM T47094 C6QD1U 9818172 IC50 > 100 nM T47094 CW1U9H 9823811 IC50 = 34.3 nM T47094 CUNL10 9824321 Ki = 4.5 nM T47094 C3WTH0 9826304 Ki = 1.288 nM T47094 C5QLA6 9827668 IC50 = 8 nM T47094 CBF5Z0 9828716 IC50 = 0.039 nM T47094 CA5M9K 9829083 IC50 = 0.85 nM T47094 CR6CG0 9830304 IC50 = 0.5 nM T47094 C1TWX8 9830535 IC50 = 41 nM T47094 CN6WE9 9831075 Ki = 1 nM T47094 CZ2EY1 9831309 IC50 = 3.1 nM T47094 C9BDV3 9831546 Ki = 0.3 nM T47094 CHIS10 9831674 Ki = 0.9 nM T47094 C3TV1U 9831707 Ki = 1.9 nM T47094 CU85VO 9832198 IC50 = 85 nM T47094 CYBE74 9832383 Ki = 0.2239 nM T47094 CKEZ38 9846661 Ki = 4.6 nM T47094 C0VED8 9846662 Ki = 8.5 nM T47094 CSA9K5 9850565 Ki = 1.7 nM T47094 CVRC05 9850771 IC50 = 0.18 nM T47094 C0RB2U 9851741 IC50 = 28 nM T47094 CIXG30 9852376 IC50 = 763 nM T47094 CMZ20K 9852630 Ki = 0.4 nM T47094 C2JS5O 9852904 Ki = 0.27 nM T47094 CTRI07 9852911 IC50 = 120 nM T47094 CSU2Y3 9853636 Ki = 0.6 nM T47094 CY37UT 9853827 Ki = 125.89 nM T47094 C9HPD2 9855000 IC50 = 0.38 nM T47094 CUND40 9868422 Ki = 17 nM T47094 C8F7ZP 9868530 IC50 = 6.1 nM T47094 CAXW26 9868622 IC50 = 23 nM T47094 C9IL0C 9869697 IC50 = 0.26 nM T47094 CAD41X 9869764 Ki = 3.4 nM T47094 CRJS21 9871414 IC50 = 0.22 nM T47094 CW13LY 9871891 IC50 = 0.21 nM T47094 CK1WO0 9872249 Ki = 1.4 nM T47094 CA3H7D 9872295 Ki = 8.128 nM T47094 CQ4LC2 9872676 Ki = 1250 nM T47094 C0YTH2 9872808 Ki = 0.2399 nM T47094 C4R3YJ 9873032 Ki = 0.44 nM T47094 C9FO1Q 9873546 IC50 = 24 nM T47094 CM3O6E 9874168 IC50 = 6.19 nM T47094 CCE74U 9874473 Ki = 0.4 nM T47094 C7W4NT 9874480 Ki = 2.512 nM T47094 CD6U7Z 9875034 Ki = 1.3 nM T47094 CA2X8G 9875056 Ki = 0.6 nM T47094 CENG46 9887525 IC50 = 2.4 nM T47094 CBT1R2 9887650 Ki = 7943.28 nM T47094 CTPD70 9888665 IC50 = 3.2 nM T47094 CY49EU 9891865 IC50 = 0.25 nM T47094 CBF3H0 9892852 IC50 = 0.2 nM T47094 C0XR2D 9892922 Ki = 10 nM T47094 CW07IY 9896757 Ki = 0.7 nM T47094 CS15YI 9910432 IC50 = 3 nM T47094 CFCG61 9916428 IC50 = 1.259 nM T47094 C4SEJ2 9917970 Ki = 0.9 nM T47094 C5U0EO 9918479 Ki = 3.3 nM T47094 C6F8RG 9918576 IC50 = 31 nM T47094 CEA1S5 9927183 IC50 = 2.399 nM T47094 CWY45T 9929728 Ki = 0.7943 nM T47094 CZ62US 9933653 IC50 = 17 nM T47094 CV5X7E 9938284 IC50 = 0.3 nM T47094 C91ZRQ 9938657 IC50 = 0.9 nM T47094 CH97DG 9939307 Ki = 4.7 nM T47094 CYRL74 9945487 IC50 = 0.41 nM T47094 C6G2OQ 9954221 IC50 = 15.14 nM T47094 CX07HS 9957036 IC50 = 700 nM T47094 C7ZXS9 9958115 Ki = 0.2 nM T47094 CWH9S8 9959330 IC50 = 1.1 nM T47094 CMGB40 9959481 IC50 > 10000 nM T47094 CZ36PE 9959724 IC50 = 0.98 nM T47094 C0DZ6K 9961315 Ki = 0.14 nM T47094 CNP82Y 9961936 Ki = 1 nM T47094 C8CY0E 9961955 Ki = 0.8 nM T47094 CM3W8D 9967131 IC50 = 0.09 nM T47094 COP51C 9968267 IC50 = 0.8 nM T47094 C5K6MJ 9976640 IC50 = 5.5 nM T47094 CY9SZ2 9978999 IC50 = 140 nM T47094 CY21QJ 9979913 IC50 = 800 nM T47094 C7FD9W 9980171 IC50 = 2.5 nM T47094 C7BG9Z 9981979 IC50 = 183 nM T47094 CP0I1O 9984184 IC50 = 56 nM T47094 CY6IM7 9984665 IC50 = 0.4 nM T47094 CIT57N 9985523 IC50 = 180 nM T47094 CO7V1Z 9987474 Ki = 14 nM T47094 CFQ13N 9988742 EC50 = 13.5 nM T47094 C7MC4I 10001148 Ki = 620 nM T47094 CZ85IN 10004377 IC50 = 0.11 nM T47094 CI89WY 10005824 IC50 = 23 nM T47094 CQP46G 10006814 IC50 = 19 nM T47094 COA65Q 10007108 Ki = 323.59 nM T47094 CG93PK 10007326 Ki = 338.84 nM T47094 CGCX36 10007758 IC50 = 0.48 nM T47094 CK56PU 10008129 IC50 = 0.3 nM T47094 C73WUR 10010039 Ki = 24 nM T47094 CZ6JW0 10010096 Ki = 6 nM T47094 C1XK9Y 10019102 IC50 > 10000 nM T47094 CH6DS8 10025594 IC50 = 760 nM T47094 CIN0Q5 10026002 IC50 = 32 nM T47094 CHZ85W 10026200 IC50 = 66 nM T47094 CU12CZ 10027061 IC50 = 25 nM T47094 CJF9Y1 10027219 IC50 = 1.5 nM T47094 CE5N2R 10027661 IC50 = 4333 nM T47094 C5ENI0 10030004 IC50 = 68 nM T47094 C3B6LV 10031310 IC50 = 7 nM T47094 CEC12Y 10032406 Ki = 9 nM T47094 C71LNR 10032693 Ki = 4 nM T47094 CVN3U7 10039383 IC50 = 1100 nM T47094 C10WEQ 10041813 IC50 = 3800 nM T47094 CGS3X5 10041814 IC50 = 1533 nM T47094 CEIQ93 10043484 IC50 = 549.54 nM T47094 CVJ8O1 10045010 IC50 = 153 nM T47094 C25WVJ 10047566 IC50 = 1 nM T47094 CU14PT 10047567 IC50 = 1 nM T47094 CRN1L3 10047989 IC50 = 280 nM T47094 CK5F4G 10049890 IC50 = 0.95 nM T47094 CY2FL7 10051762 IC50 = 0.11 nM T47094 CL78XB 10052312 IC50 = 1.2 nM T47094 C96HJL 10053174 IC50 = 0.14 nM T47094 C3L6IG 10053175 IC50 = 8.4 nM T47094 CQPM24 10053419 IC50 = 0.12 nM T47094 CF6D7J 10055415 IC50 = 165 nM T47094 CR7UY2 10063954 IC50 = 8.913 nM T47094 CW4S5I 10064734 IC50 = 1533 nM T47094 C9C0FM 10071073 IC50 = 4.4 nM T47094 C7KUO1 10071124 IC50 = 22 nM T47094 C6OI8Q 10071902 IC50 = 3600 nM T47094 CG53RU 10072926 IC50 = 4.2 nM T47094 CJP45G 10075002 IC50 = 3 nM T47094 CPF0R9 10075595 IC50 = 1.8 nM T47094 CJ6L2F 10075851 IC50 = 3.8 nM T47094 CQE8H9 10076383 IC50 = 0.65 nM T47094 CW3F4B 10076669 IC50 = 0.6 nM T47094 CQN28E 10076881 IC50 = 1.5 nM T47094 CYOC80 10077113 IC50 = 0.76 nM T47094 C25LAE 10078301 Ki = 8 nM T47094 C5D2YN 10085946 Ki = 150 nM T47094 C17EUC 10086982 IC50 = 4.2 nM T47094 C08UQI 10091563 Ki = 49 nM T47094 CB6VT4 10094248 IC50 = 19 nM T47094 CO7R9Z 10095174 IC50 = 100 nM T47094 C7F0UW 10096063 IC50 = 3.4 nM T47094 CMF7A4 10097954 IC50 = 5 nM T47094 CJQ34H 10098209 IC50 = 0.16 nM T47094 C3RJ9C 10098987 IC50 = 0.4 nM T47094 C3HA4I 10099318 IC50 = 80.9 nM T47094 C9D5FP 10099787 IC50 = 0.22 nM T47094 COL04Z 10099939 IC50 = 0.5 nM T47094 CE5NS2 10100236 IC50 = 1.7 nM T47094 CPC5B0 10101238 IC50 = 0.24 nM T47094 C1WVZ0 10102903 Ki > 10000 nM T47094 C0B6YA 10111225 IC50 = 0.14 nM T47094 CXG05H 10115747 Ki = 3.6 nM T47094 CJ2HI3 10127439 Ki = 0.7 nM T47094 CNE83S 10128086 Ki = 0.3 nM T47094 C7I3OR 10128131 Ki = 0.69 nM T47094 CQB92U 10128322 Ki = 0.3 nM T47094 CZP15C 10128366 Ki = 0.3 nM T47094 CD3E4A 10140125 Ki = 7.943 nM T47094 CT1N5S 10141196 Ki = 15.85 nM T47094 CL4IY8 10142159 IC50 = 0.78 nM T47094 CY35HP 10144275 IC50 = 0.28 nM T47094 CR1NI5 10145229 Ki = 1.8 nM T47094 C85XEY 10151946 Ki = 0.5 nM T47094 CQ9V8N 10152358 Ki = 0.29 nM T47094 CAP4T0 10152974 Ki = 0.07943 nM T47094 CQ1N8D 10164354 Ki = 0.4 nM T47094 CU81IJ 10173872 Ki = 0.1 nM T47094 CLBU87 10173890 Ki = 0.43 nM T47094 CR1G9B 10186401 IC50 = 0.15 nM T47094 CHDE36 10187704 Ki = 6.31 nM T47094 CCBF42 10189341 Ki = 18.2 nM T47094 CZCX69 10194796 Ki = 0.6 nM T47094 CT6S8X 10204249 Ki = 1.5 nM T47094 CCG65P 10210026 IC50 = 0.39 nM T47094 CSA32M 10216430 Ki = 0.02 nM T47094 CZ6C8T 10217361 Ki = 0.22 nM T47094 CGR6H7 10217362 Ki = 0.19 nM T47094 CA9XW4 10218122 Ki = 1.3 nM T47094 C9VHF5 10228092 IC50 = 41 nM T47094 CY71XB 10229773 Ki = 6.3 nM T47094 C4JW3Q 10230370 Ki = 15.85 nM T47094 CET6H5 10231172 Ki = 0.9 nM T47094 C3EC6K 10232846 Ki = 8.71 nM T47094 CQN81T 10237920 Ki = 2.4 nM T47094 CFB96H 10239000 Ki = 3.3 nM T47094 C83TKD 10239346 Ki = 1.3 nM T47094 C5KM4H 10245452 IC50 = 3500 nM T47094 CCR1F4 10251123 IC50 = 13 nM T47094 C17XLU 10253192 IC50 = 480 nM T47094 CD7NB8 10254526 IC50 = 10 nM T47094 C7ULD5 10256518 IC50 = 110 nM T47094 CYT4M9 10257218 IC50 = 0.23 nM T47094 C67GCK 10258336 IC50 = 0.63 nM T47094 CVQ23E 10258592 IC50 = 497 nM T47094 C14JSK 10258866 IC50 = 240 nM T47094 C8AG9N 10268178 IC50 = 0.46 nM T47094 C4F7IQ 10270385 Ki > 10000 nM T47094 CCF6U5 10272852 IC50 = 0.18 nM T47094 C4E0FS 10288987 Ki = 0.15 nM T47094 C1HJC9 10289302 Ki = 0.23 nM T47094 C90HVU 10290124 Ki = 0.1995 nM T47094 C7Y8HE 10295489 Ki = 6 nM T47094 CR06WO 10296442 Ki = 0.6 nM T47094 C13GVK 10299289 Ki = 8.71 nM T47094 C98XMD 10300825 Ki = 39.81 nM T47094 CBH92R 10302076 Ki = 10 nM T47094 C9HR5S 10303099 Ki = 1.12 nM T47094 CXP4Q5 10304406 Ki = 1.3 nM T47094 CN5YV6 10311126 Ki = 0.3 nM T47094 CK3N5Q 10311496 Ki = 0.59 nM T47094 C5GY4I 10317821 IC50 = 110 nM T47094 CKN9O8 10317867 IC50 = 460 nM T47094 CB8S4N 10318477 IC50 = 413 nM T47094 CT53GE 10318912 IC50 = 2632 nM T47094 C0C6KT 10318976 IC50 = 20 nM T47094 CT92GQ 10321715 Ki = 5.012 nM T47094 CWFB30 10323427 IC50 > 100 nM T47094 C4RJW3 10325464 IC50 = 420 nM T47094 CO5R8L 10325507 IC50 = 0.47 nM T47094 CF4VQ6 10327313 IC50 = 5700 nM T47094 C17NQT 10327540 IC50 = 60 nM T47094 CI5U8S 10336036 IC50 = 3700 nM T47094 C76VZT 10339539 IC50 = 7 nM T47094 CPL8J5 10341570 IC50 = 0.26 nM T47094 CK5GZ3 10342371 IC50 = 16 nM T47094 COJ4A7 10342797 IC50 = 600 nM T47094 C81FCA 10346229 IC50 = 0.33 nM T47094 CDI49K 10347274 IC50 = 0.7 nM T47094 CLN21Y 10349900 IC50 = 54 nM T47094 C1QLH0 10350241 Ki = 93000 nM T47094 CC3UG7 10350454 IC50 = 21 nM T47094 CF5M7J 10350528 IC50 = 34 nM T47094 CWO60K 10350626 IC50 > 10000 nM T47094 CP0FY4 10357939 IC50 = 0.6166 nM T47094 CN8PA7 10357986 IC50 > 10000 nM T47094 CX0E7U 10359664 IC50 = 1.995 nM T47094 CGDQ73 10360490 IC50 = 4.6 nM T47094 CZ1J0B 10362340 IC50 = 103 nM T47094 CI3YB8 10363425 IC50 = 110 nM T47094 CPW94Y 10363623 Ki = 0.3981 nM T47094 CBH35Q 10363809 IC50 = 0.11 nM T47094 CSWC08 10364638 IC50 = 19.95 nM T47094 C92BEU 10364942 IC50 = 133 nM T47094 C7SO2R 10367419 IC50 = 309.03 nM T47094 CG73OS 10369316 IC50 = 170 nM T47094 CRGN49 10369341 IC50 = 2.5 nM T47094 C0BG7R 10369373 IC50 = 0.25 nM T47094 CE64QI 10369653 IC50 = 2.8 nM T47094 C6BQR5 10369844 IC50 = 2.7 nM T47094 C9U2PN 10370593 IC50 = 54 nM T47094 CFS3N7 10370818 IC50 = 17 nM T47094 CKDL87 10372941 IC50 = 0.7 nM T47094 C20QEX 10386984 IC50 = 470 nM T47094 CJM05T 10389745 IC50 = 14 nM T47094 CYSX27 10389807 IC50 = 62 nM T47094 CU3T6J 10389968 IC50 = 11 nM T47094 CWUV34 10390130 IC50 = 6.7 nM T47094 CT9F5R 10392469 IC50 = 5.5 nM T47094 CO6Q3X 10392925 IC50 = 0.6 nM T47094 CXG7P5 10393390 IC50 = 460 nM T47094 CO9DR6 10393853 Ki = 5.129 nM T47094 C59QRY 10393962 IC50 = 0.35 nM T47094 C1AUP5 10394703 IC50 = 1.7 nM T47094 C5V0SZ 10394882 Ki = 2 nM T47094 CV5MR6 10394952 Ki = 14 nM T47094 C1IE7Y 10395141 Ki = 13 nM T47094 C4KZW9 10404051 IC50 = 433 nM T47094 C5EKJ8 10405990 IC50 = 3000 nM T47094 CTL2B7 10407571 IC50 = 16 nM T47094 C2F0AJ 10407632 IC50 = 110000 nM T47094 C8UFW9 10408564 IC50 = 860 nM T47094 CFV73Y 10408912 IC50 = 881 nM T47094 CYC91F 10409484 Ki = 95000 nM T47094 C4FQN3 10409595 IC50 = 1500 nM T47094 C49JLI 10410206 IC50 = 5500 nM T47094 CDNR80 10410322 IC50 = 5500 nM T47094 CPF5Q4 10411026 IC50 = 567 nM T47094 C7EYZ4 10412224 IC50 = 2150 nM T47094 C5AU0E 10413173 IC50 = 1.995 nM T47094 CNL13J 10414293 IC50 = 1.6 nM T47094 CJ7HS4 10414428 IC50 = 1.1 nM T47094 C71QMH 10415534 IC50 = 0.37 nM T47094 CW80YU 10415870 IC50 = 0.34 nM T47094 C9A6BX 10417108 Ki = 25 nM T47094 CDL61W 10417124 IC50 = 440 nM T47094 CNX23Q 10429546 IC50 = 138 nM T47094 C92DOU 10432488 IC50 = 32 nM T47094 CA0P2V 10433381 IC50 = 34 nM T47094 C9JPG8 10435750 IC50 = 125 nM T47094 CE5D7F 10437488 Ki = 1.259 nM T47094 COH65W 10438407 IC50 = 4.8 nM T47094 C6LXC8 10438671 IC50 = 1.5 nM T47094 C6O1GC 10439730 IC50 = 127 nM T47094 CC53GV 10441376 EC50 = 14 nM T47094 CNEW69 10448006 IC50 = 2333 nM T47094 C0OK8L 10451098 IC50 = 6700 nM T47094 CE4X3S 10453364 IC50 = 34 nM T47094 CN9W2K 10454303 IC50 = 840 nM T47094 CH7F6K 10456592 IC50 = 28 nM T47094 CH1S7N 10456618 IC50 = 203 nM T47094 C6LS3A 10457416 IC50 = 2.2 nM T47094 CD8CE4 10458783 IC50 = 227 nM T47094 CY8I2T 10458786 IC50 = 600 nM T47094 C60BHZ 10459262 IC50 = 250 nM T47094 CP9HD4 10460415 IC50 = 4.6 nM T47094 CZH57O 10460917 IC50 = 0.1698 nM T47094 CYDW30 10462250 IC50 = 1.8 nM T47094 CS57CU 10474902 IC50 = 87 nM T47094 C3TU4X 10476340 Ki = 0.7943 nM T47094 CW4S1G 10476776 IC50 = 30 nM T47094 C31BTI 10477667 IC50 > 100 nM T47094 CY07LB 10477952 IC50 = 1050 nM T47094 CTFZ13 10477953 IC50 = 243 nM T47094 CO49AP 10478708 IC50 = 2400 nM T47094 C72FKI 10480465 IC50 = 0.1995 nM T47094 C91QYL 10480944 IC50 = 31 nM T47094 C21CWX 10483816 IC50 = 0.34 nM T47094 CO6VE5 10484232 IC50 = 23 nM T47094 CN9WY7 10484667 Ki = 20 nM T47094 C2XC3N 10495476 Ki = 0.1585 nM T47094 CSQK61 10499614 Ki = 0.0631 nM T47094 CEW41X 10499624 IC50 = 55 nM T47094 CLJ4I6 10499846 IC50 = 90 nM T47094 CYNX98 10500669 Ki = 0.05012 nM T47094 C5CZK6 10501444 IC50 = 376 nM T47094 CXKM90 10502796 IC50 = 0.7 nM T47094 C6L7IK 10503457 IC50 > 50000 nM T47094 C6C0HY 10506124 IC50 = 270 nM T47094 CX8VP1 10506376 IC50 = 21.9 nM T47094 CD6G1Q 10506928 IC50 = 358 nM T47094 CNB0S4 10506929 IC50 = 2.5 nM T47094 CWIN19 10507650 Ki = 3.8 nM T47094 CN5HT3 10507771 Ki = 17.1 nM T47094 CCM1B9 10507772 Ki = 36 nM T47094 CXPO50 10520658 IC50 = 2933 nM T47094 C5QRF4 10522676 Ki = 0.5012 nM T47094 C40NYC 10529338 IC50 = 1.8 nM T47094 CYV94J 10530317 IC50 = 590 nM T47094 C8PJG0 10530375 Ki = 0.88 nM T47094 CU51SG 10530444 IC50 = 126 nM T47094 CEL1V5 10530592 Ki = 260 nM T47094 C8CZ4H 10530699 IC50 = 3.1 nM T47094 C1JDZ2 10530741 Ki = 3.5 nM T47094 C52XGL 10531050 IC50 = 0.98 nM T47094 C7L3FX 10531273 Ki = 172 nM T47094 CY5C6R 10531291 IC50 = 160 nM T47094 C96JKO 10531434 Ki = 16.7 nM T47094 CYP97F 10531588 IC50 = 9.2 nM T47094 CLI25C 10531666 Ki = 4.7 nM T47094 CQ3U6W 10533328 IC50 = 1389 nM T47094 C8XAF3 10533610 IC50 = 59 nM T47094 C3C2ZQ 10546738 Ki = 0.1259 nM T47094 C39KAJ 10547681 Ki = 0.1995 nM T47094 CNX09U 10548166 IC50 = 84 nM T47094 CV59GA 10552574 IC50 = 33 nM T47094 CG04NV 10552836 IC50 = 36 nM T47094 CDS3H9 10553136 IC50 = 5.3 nM T47094 CA4C3D 10553717 IC50 > 5000 nM T47094 C0IJ6L 10553958 IC50 = 300 nM T47094 C46RBI 10553959 IC50 = 0.2 nM T47094 CNL4C3 10554361 IC50 = 1.8 nM T47094 COZ8Y1 10555763 Ki = 1.7 nM T47094 CLV51H 10556941 IC50 = 209 nM T47094 CP6U3T 10557646 IC50 = 2 nM T47094 C3T8QH 10572904 IC50 > 1000 nM T47094 C86DOM 10573735 IC50 > 1000 nM T47094 CJWN14 10576865 IC50 = 0.97 nM T47094 CJ8Y1K 10576866 IC50 = 39.81 nM T47094 C1VGZ6 10577745 IC50 = 8.3 nM T47094 C58EHT 10578261 Ki = 6.7 nM T47094 C96RTO 10578269 IC50 = 0.94 nM T47094 C8OE3N 10578351 IC50 = 0.8 nM T47094 CO8IX4 10578969 IC50 = 1.18 nM T47094 CHM8Q1 10581337 IC50 = 198 nM T47094 CH3F1E 10599370 IC50 > 50000 nM T47094 C7H2VK 10600014 Ki = 330 nM T47094 C6FI2Y 10600310 Ki = 2.8 nM T47094 CJ2G3D 10601035 IC50 > 50000 nM T47094 CF4IP1 10602065 IC50 = 6.9 nM T47094 CO3DB5 10602943 Ki = 4.2 nM T47094 C42UCR 10603019 IC50 = 2.73 nM T47094 CE35HF 10603097 IC50 = 3 nM T47094 C3SX0I 10603279 Ki = 5 nM T47094 CAX58F 10603365 Ki = 27.2 nM T47094 CL3D1S 10603383 Ki = 25.9 nM T47094 CB2RM1 10603392 IC50 = 5.5 nM T47094 CN9SC8 10603544 Ki = 0.3 nM T47094 C8UEI1 10619783 Ki > 100000 nM T47094 C2K7RE 10620143 IC50 = 57 nM T47094 CQF79S 10621261 Ki = 0.7943 nM T47094 CXW2U5 10621581 IC50 > 1000 nM T47094 CL6VD2 10623161 IC50 > 50000 nM T47094 C3XVR5 10623791 IC50 = 5.3 nM T47094 CXEY42 10624321 IC50 > 50000 nM T47094 CDF3Y2 10624372 IC50 = 2.8 nM T47094 CK91JP 10625208 IC50 = 474 nM T47094 C31GJT 10626048 IC50 = 1.2 nM T47094 C8KNR1 10626666 Ki = 1.1 nM T47094 C9M2XG 10626865 IC50 = 7.2 nM T47094 CV41GB 10627355 IC50 = 1.54 nM T47094 C6FSM5 10627789 Ki = 27 nM T47094 C4ZGL1 10641076 Ki = 0.07943 nM T47094 CD4M3N 10643148 Ki = 0.1585 nM T47094 CL4J9F 10646925 IC50 = 38 nM T47094 CTN8U2 10648288 IC50 = 1.6 nM T47094 CI1HS7 10648551 IC50 = 1 nM T47094 C0K7FQ 10649307 Ki = 1700 nM T47094 CE4WO8 10649931 Ki = 18.5 nM T47094 C91FUP 10649948 IC50 = 290 nM T47094 C8SAY7 10650469 IC50 = 1.9 nM T47094 CNTC13 10650495 Ki = 1.1 nM T47094 C5YM1V 10651193 Ki = 13.7 nM T47094 CYO80C 10651575 Ki = 7.2 nM T47094 CLOF45 10668461 Ki > 100000 nM T47094 CY0IO7 10668476 IC50 = 700 nM T47094 CS9C3X 10669293 IC50 = 2.9 nM T47094 C1XB2T 10670029 IC50 > 5000 nM T47094 CH3V2U 10671119 IC50 > 5000 nM T47094 C5SXF6 10671903 IC50 > 5000 nM T47094 C02YTI 10672166 IC50 > 5000 nM T47094 C7WM4G 10674548 IC50 = 3 nM T47094 C7N9JL 10674743 IC50 = 7100 nM T47094 C1SOY6 10675169 Ki = 6.1 nM T47094 CZ1K3M 10691318 Ki > 100000 nM T47094 C6P9UI 10692651 IC50 = 59 nM T47094 CA0T8Y 10695397 IC50 = 66 nM T47094 C4JA2Q 10696382 IC50 = 3.1 nM T47094 CYT13I 10697072 IC50 = 51 nM T47094 C0N2YH 10697884 Ki = 29.9 nM T47094 CGP7A5 10698085 IC50 = 9.5 nM T47094 CDC7Q5 10698096 IC50 = 0.34 nM T47094 C15TCW 10698161 IC50 = 206 nM T47094 C8IR7A 10698493 Ki = 0.5 nM T47094 C3SU0I 10698708 Ki = 29.7 nM T47094 CB4NM8 10700731 IC50 = 28 nM T47094 C1R0MF 10714695 Ki = 0.03162 nM T47094 CH64RI 10720240 IC50 = 0.5 nM T47094 C40LWB 10721128 IC50 = 3.2 nM T47094 C73NFE 10721713 IC50 = 0.81 nM T47094 C0FT3Z 10722491 IC50 = 2 nM T47094 CZS4R3 10722607 Ki = 29.4 nM T47094 CEFN53 10723865 IC50 = 596 nM T47094 CU2K1T 10736544 IC50 = 750 nM T47094 CJ1B7C 10743826 IC50 = 5.7 nM T47094 CL1ES4 10744602 IC50 = 2.2 nM T47094 CW5R4K 10744740 IC50 = 410 nM T47094 C24MHU 10744888 IC50 = 100000 nM T47094 C3U5DL 10745123 Ki = 1280 nM T47094 C7GH4X 10745241 IC50 = 19700 nM T47094 C8ZN4E 10745307 IC50 = 4.6 nM T47094 CN9H1R 10745532 Ki = 1.7 nM T47094 CP6FB5 10745788 IC50 = 274000 nM T47094 C4FWO2 10746177 Ki = 18.2 nM T47094 C32MYS 10746828 Ki = 78.6 nM T47094 C4FN1T 10748217 IC50 = 15 nM T47094 C1QI4M 10761962 Ki = 0.5012 nM T47094 C8GZ4A 10763310 IC50 > 1000 nM T47094 CJP9Z1 10764172 IC50 > 1000 nM T47094 CN8L6T 10766356 IC50 > 5000 nM T47094 C5P8NB 10767359 IC50 = 149 nM T47094 CD4BG9 10767720 Ki = 80 nM T47094 CS5QP8 10768417 IC50 = 0.32 nM T47094 CK8UI4 10769059 Ki = 0.7 nM T47094 CR0W8S 10769060 Ki = 2.2 nM T47094 CJW85Q 10769264 IC50 = 2500 nM T47094 CQIY49 10769745 IC50 = 3.2 nM T47094 C84LDO 10769914 Ki = 48 nM T47094 CB97OQ 10784942 Ki = 0.1585 nM T47094 CHFQ21 10788622 IC50 > 1000 nM T47094 CPF8E2 10790280 Ki = 170 nM T47094 C8C9XJ 10790827 IC50 = 27 nM T47094 COY96S 10792813 IC50 = 4.5 nM T47094 C4TJF0 10792994 Ki = 8000 nM T47094 C0U8XG 10793140 IC50 = 338 nM T47094 C14TVO 10793340 Ki = 2.3 nM T47094 CMF58R 10793341 IC50 = 1000 nM T47094 C24AKU 10793492 IC50 = 3700 nM T47094 CUFS78 10793838 IC50 = 1.28 nM T47094 C3MZ4I 10794699 Ki = 26.9 nM T47094 CJI56W 10795155 IC50 = 4093 nM T47094 CHP78E 10795384 IC50 = 2732 nM T47094 CUO64P 10809458 Ki = 0.05012 nM T47094 C72ITB 10811257 IC50 = 21 nM T47094 C5X1LM 10812646 IC50 > 1000 nM T47094 CC1W4K 10813332 Ki = 1270 nM T47094 C0P2YR 10814682 IC50 = 0.53 nM T47094 CZY2F4 10815815 IC50 = 2.8 nM T47094 CM5A1X 10816374 IC50 = 0.85 nM T47094 C3S5VU 10816496 Ki = 2.6 nM T47094 CN6FA4 10816935 IC50 = 1.8 nM T47094 CI5BV1 10817013 Ki = 0.8 nM T47094 CO02AJ 10817098 Ki = 2.3 nM T47094 C8DI7P 10817203 IC50 = 4 nM T47094 CDJ2M8 10817360 Ki = 0.7 nM T47094 CG9TH3 10819275 IC50 = 216 nM T47094 CF8OS4 10834119 IC50 = 2.4 nM T47094 C7IV9Y 10834930 IC50 = 170 nM T47094 C2G8RZ 10835447 IC50 = 1700 nM T47094 CNB3U8 10836352 IC50 > 5000 nM T47094 CDTN64 10837320 IC50 = 63 nM T47094 CR0T2Y 10837362 IC50 = 12.6 nM T47094 CE2UP1 10837611 IC50 = 2.9 nM T47094 CC0MB6 10837742 IC50 = 1.1 nM T47094 CEKX50 10837983 IC50 > 50000 nM T47094 CS3T9C 10839068 IC50 = 7.3 nM T47094 CFB30H 10839138 Ki = 220 nM T47094 C9X3GQ 10840066 IC50 = 1.8 nM T47094 CG6ZB8 10840161 IC50 = 85 nM T47094 CCK38X 10840399 IC50 = 10000 nM T47094 C14LFR 10840510 IC50 = 27.4 nM T47094 CBO2I1 10840688 IC50 = 11 nM T47094 CP69MV 10841047 IC50 = 31 nM T47094 CV1CW0 10885893 IC50 = 0.7 nM T47094 CX65PW 10907460 IC50 = 839 nM T47094 C4SBO9 10915140 IC50 > 10000 nM T47094 C3X5FP 10951720 IC50 = 0.25 nM T47094 CTA6Q1 11016806 IC50 = 0.85 nM T47094 C9CQ8N 11114226 IC50 = 3.79 nM T47094 C0IB6Y 11146618 IC50 = 0.35 nM T47094 CCN14J 11156351 IC50 = 0.0017 nM T47094 CF8DK1 11192771 IC50 = 180 nM T47094 C3DA9X 11225834 IC50 = 3.1 nM T47094 C8YQ6F 11238415 IC50 = 0.01 nM T47094 CAB10S 11239751 Ki = 199.53 nM T47094 C3DI1T 11248796 IC50 = 0.03 nM T47094 C52CJT 11261795 Ki = 0.537 nM T47094 C2TC9K 11273015 Ki = 130 nM T47094 CWM7X9 11295303 IC50 = 9 nM T47094 CZ90JO 11296094 Ki = 0.78 nM T47094 C08OTJ 11305162 Ki = 51 nM T47094 C7YA4O 11318556 IC50 = 11 nM T47094 CL68HC 11325534 IC50 > 100000 nM T47094 CW6O0E 11327981 IC50 < 0.1 nM T47094 COJE81 11329897 IC50 = 26 nM T47094 C3FVB2 11352855 IC50 = 0.011 nM T47094 CN9B1I 11353915 Ki = 2.24 nM T47094 CW43YL 11363490 IC50 = 208 nM T47094 CG1N5H 11399132 IC50 > 1000 nM T47094 CO5FQ6 11399458 IC50 > 1000 nM T47094 CX6GP2 11409185 IC50 = 0.075 nM T47094 C5PG2E 11433531 IC50 = 17 nM T47094 CAQ2N7 11445389 IC50 = 12000 nM T47094 C8Z9SV 11467400 Ki = 3.37 nM T47094 CM7BZ8 11475738 Ki > 10000 nM T47094 CEA14U 11489240 IC50 = 16 nM T47094 C2O8ER 11489471 IC50 = 11 nM T47094 CDC01U 11490127 IC50 = 52 nM T47094 C5USE7 11490769 Ki = 0.4 nM T47094 C21EUP 11497630 IC50 > 100 nM T47094 CSM9N1 11518191 IC50 = 16 nM T47094 CE7KD1 11539564 IC50 = 2.6 nM T47094 C0AP8I 11546190 IC50 = 7.5 nM T47094 CUQ3H4 11546759 IC50 = 7.2 nM T47094 C8VB1F 11547090 IC50 = 32 nM T47094 CQ74AN 11547594 IC50 = 4.7 nM T47094 CJ1YS8 11561036 IC50 = 2.6 nM T47094 COR0D7 11568372 IC50 = 1.4 nM T47094 CN78BY 11612528 IC50 = 14 nM T47094 CI63EU 11619202 IC50 = 6.7 nM T47094 C68QNP 11621512 IC50 = 0.047 nM T47094 CEZJ35 11633082 IC50 = 19 nM T47094 CQX2N5 11634999 IC50 = 74 nM T47094 CU9AE6 11641636 IC50 = 45 nM T47094 CGD21T 11642147 IC50 = 26 nM T47094 C8T9RB 11647974 IC50 = 8 nM T47094 CM2E6F 11654898 IC50 = 2.5 nM T47094 C51BJP 11661466 IC50 = 950 nM T47094 C50QHI 11661655 IC50 = 31 nM T47094 C34RDZ 11678857 IC50 = 0.33 nM T47094 CZHQ32 11683136 IC50 = 11 nM T47094 CJ20GB 11705241 IC50 = 11 nM T47094 CJ53MI 11705830 IC50 = 20 nM T47094 C8GO3J 11712457 Ki = 0.3 nM T47094 CPKL94 11723662 Ki < 1000 nM T47094 CN3ME8 11724403 IC50 = 120 nM T47094 C1E7TL 11734825 Ki = 0.8318 nM T47094 CCG0F7 11743207 IC50 = 16 nM T47094 CYU45Z 11743365 IC50 = 5.1 nM T47094 C4YL8Z 11755227 IC50 = 0.3 nM T47094 CSQ5L1 11755361 IC50 = 1.905 nM T47094 CKO04S 11756257 IC50 = 0.43 nM T47094 CZX6M8 11756817 IC50 > 100 nM T47094 CV97HR 11756839 IC50 = 1.3 nM T47094 CO5IL2 11757401 IC50 = 2 nM T47094 CQAY15 11793012 Ki = 0.0631 nM T47094 CBF81P 11793946 Ki = 1.995 nM T47094 CR5W1U 11794060 Ki = 2.512 nM T47094 CDT39Q 11799022 IC50 = 0.9 nM T47094 CV58YE 11799987 Ki = 1010 nM T47094 CJ6HG7 11800024 IC50 = 0.7943 nM T47094 C1WKM0 11800025 IC50 = 0.6 nM T47094 CWU0V1 11800372 IC50 = 2.3 nM T47094 CHR0C1 11801041 Ki = 38 nM T47094 C1A2RO 11801327 Ki = 1 nM T47094 CM24FX 11801586 IC50 = 9600 nM T47094 C4ARI6 11801965 Ki = 5 nM T47094 CU28DZ 11803184 IC50 = 549 nM T47094 CI14KO 11803645 IC50 = 1045 nM T47094 CJ2HF8 11813209 IC50 = 0.96 nM T47094 C40ABD 11814040 IC50 = 0.21 nM T47094 C2J8RH 11844212 IC50 = 50 nM T47094 CTJK89 11852872 IC50 = 0.073 nM T47094 C1O8ZJ 11983278 IC50 = 0.09 nM T47094 C0D3JE 12047485 IC50 = 165 nM T47094 C0Q4EW 12096357 IC50 = 159 nM T47094 CZO54M 14986134 IC50 = 3.4 nM T47094 C8VX6O 14986135 IC50 = 0.33 nM T47094 CN5KR2 15214194 IC50 = 3.4 nM T47094 CFPY12 15253734 IC50 = 0.18 nM T47094 CW06TB 15295987 IC50 = 400 nM T47094 C2HI3O 15295988 IC50 = 243 nM T47094 C6C1QB 15295989 IC50 = 267 nM T47094 CE01FG 15391369 IC50 = 68 nM T47094 C0OU2J 15485361 IC50 = 1026 nM T47094 COJ24C 15508105 Ki = 1.2 nM T47094 COT10M 15516313 IC50 = 0.34 nM T47094 C4FY2P 15549736 IC50 < 0.1 nM T47094 C21ITW 15549737 IC50 = 0.9 nM T47094 C4IT0Z 15639102 IC50 = 169.82 nM T47094 CE5I9T 15639109 IC50 = 67.61 nM T47094 C92PML 15639110 IC50 = 0.912 nM T47094 C3ETC8 15639130 IC50 = 229.09 nM T47094 CQI15J 15639149 IC50 = 1.905 nM T47094 CN8XO4 15887536 Ki = 136 nM T47094 C8N2EM 15887537 Ki = 5.3 nM T47094 CDZ0X9 16006943 IC50 = 0.16 nM T47094 C4SOQ7 16214865 IC50 = 146 nM T47094 C0CRS4 16663280 IC50 = 0.06 nM T47094 CG9WC1 16735704 Ki = 3 nM T47094 C20SRH 16737292 Ki = 0.88 nM T47094 C9GZ7X 16737294 Ki = 1 nM T47094 C9MZD1 16737629 Ki = 0.8 nM T47094 C0EBA3 16737631 Ki = 0.2 nM T47094 C23MPB 16737673 Ki = 0.082 nM T47094 CR7X1S 16755206 IC50 = 390 nM T47094 C80YHR 16755228 IC50 = 36 nM T47094 CCVP01 16755229 IC50 = 1233 nM T47094 C6ZUO2 16755230 IC50 = 38 nM T47094 CCH17I 16755231 IC50 = 4.3 nM T47094 CVNQ68 16755232 IC50 = 542 nM T47094 C5C7MD 16755253 IC50 = 9 nM T47094 CU83BN 16755254 IC50 = 311 nM T47094 CBHR16 16755255 IC50 = 26 nM T47094 C2IO3R 16755256 IC50 = 401 nM T47094 CDZ1L6 16755257 IC50 = 55 nM T47094 CYR81P 16755278 IC50 = 235 nM T47094 CC0SM4 16755279 IC50 = 21 nM T47094 C6W4FV 16755280 IC50 = 2749 nM T47094 C4AP2I 16755281 IC50 = 780 nM T47094 CXT42P 18391045 IC50 = 10 nM T47094 CN38IK 18391053 IC50 = 62 nM T47094 CA3SL9 18393120 Ki = 215 nM T47094 C7ADZ9 18403344 Ki = 0.4 nM T47094 CS90LJ 18407037 IC50 = 0.28 nM T47094 CAW9P5 18407045 IC50 = 2.6 nM T47094 CIR76A 18546495 Ki = 562 nM T47094 CTL13E 18546500 Ki = 224 nM T47094 CLI85K 18654560 IC50 = 290 nM T47094 CR04UX 18654565 IC50 = 17 nM T47094 CY2B6R 18655106 IC50 = 500 nM T47094 CB68ZA 18667231 Ki = 0.2512 nM T47094 C5J9IG 18669055 IC50 = 2 nM T47094 CC18FK 18669059 IC50 = 0.44 nM T47094 C0GM6D 18669072 IC50 = 0.97 nM T47094 C5CZU7 18669080 IC50 = 0.39 nM T47094 CZ37RH 18669082 IC50 = 0.6 nM T47094 C7KBJ1 18669085 IC50 = 7.6 nM T47094 CP0UL9 18669087 IC50 = 0.89 nM T47094 CBY0F8 18669089 IC50 = 6.3 nM T47094 CF40DB 18669091 IC50 = 0.3 nM T47094 CHV0J2 18669097 IC50 = 0.2 nM T47094 C1N8TD 18686789 IC50 = 0.61 nM T47094 CR2VE5 18709628 IC50 = 24 nM T47094 CK6D8G 18709649 IC50 = 0.82 nM T47094 C7H4AK 18709650 IC50 = 3.2 nM T47094 CRI7U6 18709652 IC50 = 10.2 nM T47094 C9IA2L 18709663 IC50 = 3.5 nM T47094 CXW06B 18782542 IC50 = 0.35 nM T47094 CZO30N 18782568 IC50 = 49 nM T47094 CYVI40 18986937 IC50 = 80 nM T47094 CZ4U1J 18986942 IC50 = 93 nM T47094 C0BI9O 19003143 IC50 = 2333 nM T47094 C5QO9S 19003156 IC50 = 67 nM T47094 C3TUO5 19003165 IC50 = 1160 nM T47094 CNL37J 19003169 IC50 = 483 nM T47094 CIB3Q7 19049319 IC50 = 9.3 nM T47094 C09LTM 19049350 IC50 = 10.7 nM T47094 C7ITE2 19098236 IC50 = 7.5 nM T47094 CZ8I5Y 19098237 IC50 = 3.9 nM T47094 CCG67R 19610193 Ki = 112 nM T47094 CSCH45 19797413 IC50 = 33 nM T47094 CQT7R2 19797414 IC50 = 93 nM T47094 CKTI17 19797415 IC50 = 62 nM T47094 CC8QE5 19797417 IC50 = 80 nM T47094 CV31AP 19797419 IC50 = 20 nM T47094 CZL4Y3 19797420 IC50 = 300 nM T47094 C4UGV8 19797422 IC50 = 0.32 nM T47094 CIF03J 19797425 IC50 = 172 nM T47094 CEIQ65 19797429 IC50 = 197 nM T47094 C9UTM1 19797431 IC50 = 252 nM T47094 CWF73O 19797432 IC50 = 1.5 nM T47094 C3IY6E 19797436 IC50 = 37 nM T47094 CXU2T9 19797439 IC50 = 8.3 nM T47094 C0FL4J 19797443 IC50 = 127 nM T47094 CGK2O1 19797445 IC50 = 86 nM T47094 C1IUT7 19797446 IC50 = 370 nM T47094 C9UK4S 19797448 IC50 = 37 nM T47094 C1PKX6 19797451 IC50 = 246 nM T47094 C3HD6J 19797452 IC50 = 1113 nM T47094 CU26YN 19797456 IC50 = 36 nM T47094 CDIF13 19797458 IC50 = 62 nM T47094 C7VPX5 19797460 IC50 = 9 nM T47094 C7QUT3 19797466 IC50 = 417 nM T47094 C05OVM 19797468 IC50 = 67 nM T47094 CF85JR 19797472 IC50 = 0.9 nM T47094 CM2P7J 19797474 IC50 = 106 nM T47094 C61VJE 19797477 IC50 = 56 nM T47094 CY6HT9 19797480 IC50 = 150 nM T47094 CQY49J 19960248 IC50 = 730 nM T47094 CC86AS 19968650 IC50 = 13.5 nM T47094 CKT39N 20599010 Ki = 6.31 nM T47094 C8KZ4Y 20599018 Ki = 1.259 nM T47094 CG5JB7 20811360 Ki = 7.943 nM T47094 C81JWV 20906619 Ki = 1800 nM T47094 CI9D8J 21041073 Ki = 0.1995 nM T47094 CMA0D8 21050485 IC50 = 1.6 nM T47094 C6ZQC4 21121353 IC50 = 6 nM T47094 CF45EV 21256636 IC50 = 280 nM T47094 CBPR58 21308488 IC50 = 547 nM T47094 C01MKX 21308490 IC50 = 602 nM T47094 C0DM3V 21753663 IC50 = 11 nM T47094 CJR06T 21753665 IC50 = 21 nM T47094 CJ53PS 21955222 IC50 = 0.49 nM T47094 CTQ5O3 21955285 IC50 = 0.44 nM T47094 CTAH93 21955298 IC50 = 0.7 nM T47094 CU0O4K 21955317 IC50 = 0.33 nM T47094 CFKU92 21994241 IC50 = 850 nM T47094 C9A6BF 21994258 IC50 = 3.3 nM T47094 CF0T6Y 21994270 IC50 = 19 nM T47094 C5B7ZP 21994307 IC50 = 1.6 nM T47094 CU9I2D 21994308 IC50 = 270 nM T47094 CV65BA 21994327 IC50 = 2.8 nM T47094 CG0MO7 21994328 IC50 = 7 nM T47094 C48DEJ 21994329 IC50 = 61 nM T47094 CEK5F8 21994340 IC50 = 2.3 nM T47094 CY3Z7A 21994346 IC50 = 2400 nM T47094 C31DQS 21994352 IC50 = 7.2 nM T47094 CP04TB 21994362 IC50 = 2200 nM T47094 COD2Q5 21994363 IC50 = 250 nM T47094 CT4X5K 21994365 IC50 = 15 nM T47094 CLN9C7 22000062 Ki = 3.3 nM T47094 CFZ7U4 22293463 IC50 = 5.3 nM T47094 CYM05F 22293473 IC50 = 120 nM T47094 CBY02H 22293475 IC50 = 0.35 nM T47094 CRC8H3 22293476 IC50 = 1.7 nM T47094 CN1O7Z 22293490 IC50 = 0.29 nM T47094 C4A1EI 22293505 IC50 = 0.75 nM T47094 CB8G5H 22293526 IC50 = 6.3 nM T47094 C08RCN 22293565 IC50 = 2.5 nM T47094 C4UXK9 22293578 IC50 = 40 nM T47094 C4X8WL 22353151 Ki = 1.585 nM T47094 CFX6E0 22353158 Ki = 1.995 nM T47094 CEB1M3 22724580 IC50 = 3 nM T47094 CI15KP 22850669 IC50 = 130 nM T47094 C3MK7H 22851562 IC50 = 540 nM T47094 C0LR3P 22859115 IC50 = 13 nM T47094 CS9E4H 22859118 IC50 = 23 nM T47094 CP2EW9 22869971 IC50 = 180 nM T47094 C0DSR9 22879211 IC50 = 0.56 nM T47094 CHQ5M2 22880694 Ki = 0.03981 nM T47094 CW1IN0 22880698 Ki = 0.3981 nM T47094 CF9LA0 22880715 Ki = 0.07943 nM T47094 CU0P3T 22880718 Ki = 0.0631 nM T47094 CFEG67 22885615 IC50 = 0.17 nM T47094 C6F1CQ 22885690 IC50 = 1.3 nM T47094 CTSI69 22885691 IC50 = 0.25 nM T47094 CP9Q0R 22885692 IC50 = 0.25 nM T47094 C26KSO 22885694 IC50 = 0.14 nM T47094 C09YOF 22885695 IC50 = 0.3 nM T47094 CP52YC 22885696 IC50 = 0.34 nM T47094 CK61WX 22885697 IC50 = 0.2 nM T47094 CHOG80 22885698 IC50 = 0.24 nM T47094 CKIR74 22885699 IC50 = 0.19 nM T47094 CPA47O 22885702 IC50 = 0.39 nM T47094 CI5T3U 22885703 IC50 = 0.19 nM T47094 CVNW27 22885704 IC50 = 0.38 nM T47094 CA9KU2 22901329 IC50 = 0.53 nM T47094 CV71IN 22960738 Ki = 0.4 nM T47094 CVXM39 22960739 Ki = 1.6 nM T47094 CD36LE 23025460 IC50 = 5.9 nM T47094 CX2DE3 23025476 IC50 = 97 nM T47094 C6IV2L 23025481 IC50 = 2.6 nM T47094 C8RL0T 23146876 IC50 = 0.17 nM T47094 CXF8Z9 23294208 IC50 = 743 nM T47094 C3XN1D 23294214 IC50 = 379 nM T47094 CMB2Z1 24180495 IC50 = 0.07 nM T47094 C57DJQ 24750734 IC50 = 0.09 nM T47094 C6ZA9Y 24750888 IC50 = 0.42 nM T47094 CM2LI5 24752434 IC50 = 0.91 nM T47094 C3S8NH 24752568 IC50 = 0.38 nM T47094 CS09VF 24752718 IC50 = 0.05 nM T47094 CJ8Q4N 24755076 IC50 = 0.22 nM T47094 CEF65A 24768357 Ki = 0.6 nM T47094 CN3AY8 24768358 Ki = 0.71 nM T47094 C3P7IS 24768572 IC50 = 0.18 nM T47094 CO8IA7 24785717 IC50 = 0.2 nM T47094 C4JK2Q 24785978 IC50 = 0.59 nM T47094 CDQ58K 24799187 IC50 = 6.3 nM T47094 CTQ59S 24799364 IC50 = 3 nM T47094 C8LJY2 24799365 IC50 = 760 nM T47094 CO32ND 24799366 IC50 = 1.6 nM T47094 C6X0JS 24799545 IC50 = 1 nM T47094 CG24KB 24799546 IC50 = 180 nM T47094 C1QL3V 24799711 IC50 = 22 nM T47094 CH0Y9J 24800231 IC50 = 1.9 nM T47094 C10YFG 24800398 IC50 = 6.1 nM T47094 C3FYB5 24800577 IC50 = 790 nM T47094 C17RDK 24800578 IC50 = 2.7 nM T47094 C30UAB 24800743 IC50 = 20 nM T47094 C6SHG9 24800925 IC50 = 600 nM T47094 C0L6CF 24800927 IC50 = 11 nM T47094 CM2K4N 24801101 IC50 = 29 nM T47094 CP8T1L 24801102 IC50 = 34 nM T47094 CA8GT1 24801457 IC50 = 45 nM T47094 CW8GD6 24801458 IC50 = 1.2 nM T47094 CE25UP 24801459 IC50 = 380 nM T47094 CSK49W 24801626 IC50 = 12 nM T47094 C1NK4A 24801627 IC50 = 66 nM T47094 C9GK5S 24801792 IC50 = 52 nM T47094 CWH29M 24801795 IC50 = 13 nM T47094 C84TEM 24801797 IC50 = 29 nM T47094 CH25PW 24888772 IC50 = 0.14 nM T47094 C1V5PM 24888942 IC50 = 0.18 nM T47094 C52QPN 24888943 IC50 = 0.09 nM T47094 COMH90 24889111 IC50 = 1 nM T47094 C45DMO 24889113 IC50 = 0.066 nM T47094 CARY25 24889114 IC50 = 0.15 nM T47094 C63SEW 24889283 IC50 = 1.7 nM T47094 CHIQ64 24889458 IC50 = 0.4 nM T47094 C3C0KP 24894134 EC50 > 50000 nM T47094 CO69SF 24969015 Ki = 0.06457 nM T47094 CL32KM 24969353 Ki = 0.5012 nM T47094 CT5QM3 24992986 IC50 = 0.255 nM T47094 CC93WO 24993312 IC50 = 0.15 nM T47094 CC1KG8 24993313 IC50 = 0.09 nM T47094 CK56YD 24993314 IC50 = 0.1 nM T47094 C0KP1S 24993955 IC50 = 7.8 nM T47094 CQ6RB4 25027805 IC50 = 0.017 nM T47094 CEI9L2 25129133 Ki = 0.0065 nM T47094 C0YOQ7 25176461 IC50 = 2 nM T47094 C1JL9X 25176462 IC50 = 2 nM T47094 C08BLI 25221995 Ki = 181.6 nM T47094 C3VJ0E 25222441 Ki = 151.8 nM T47094 C0Q2WD 28558057 IC50 = 6561 nM T47094 C18EYP 40727876 IC50 = 6.5 nM T47094 CHFX96 42639649 IC50 = 0.525 nM T47094 CDF13E 42639650 IC50 = 0.13 nM T47094 CVP9I0 44138555 Ki = 3.715 nM T47094 C1XGJ4 44138558 Ki = 18.2 nM T47094 C0KZG4 44140365 Ki = 0.4266 nM T47094 CU0PY1 44176456 Ki = 0.12 nM T47094 C7DR0P 44176458 Ki = 0.004 nM T47094 C4ZS5G 44176572 Ki = 0.03 nM T47094 CP0WQ3 44177145 IC50 = 0.002692 nM T47094 CHJ47Y 44177567 Ki = 0.034 nM T47094 C1W9PD 44177570 Ki = 0.075 nM T47094 CHI47S 44177668 Ki = 0.12 nM T47094 C2E1GB 44177669 Ki = 0.21 nM T47094 CD3LH2 44177670 Ki = 1 nM T47094 CX2O9F 44177768 Ki = 0.88 nM T47094 C8XDQ3 44177770 Ki = 0.05 nM T47094 CPHW46 44177994 Ki = 0.009 nM T47094 CHAO36 44177995 Ki = 0.09 nM T47094 CVOJ62 44178113 Ki = 0.0079 nM T47094 CANJ87 44212281 IC50 = 22.8 nM T47094 CJV13F 44212282 IC50 = 73.6 nM T47094 CBFR56 44212283 IC50 = 48.2 nM T47094 C0WQ8T 44212284 IC50 = 127 nM T47094 C1TNM2 44212285 IC50 = 271 nM T47094 CU1SX2 44212684 IC50 = 226 nM T47094 CY9MG6 44212688 IC50 = 2235 nM T47094 C1UCG8 44213477 IC50 = 170 nM T47094 C46PEF 44215303 Ki = 13 nM T47094 C16DHL 44215305 Ki = 10 nM T47094 CB4CJ8 44215306 Ki = 13 nM T47094 C73ILF 44216236 Ki = 1.15 nM T47094 CF26JI 44233184 Ki = 1.8 nM T47094 C67CEB 44233185 Ki = 0.077 nM T47094 CSB84Q 44233410 IC50 = 0.0006166 nM T47094 CO9N0V 44241710 Ki = 0.7 nM T47094 CRQB98 44241723 Ki = 0.3 nM T47094 CP37XK 44266422 Ki > 100000 nM T47094 C0WK7U 44266459 Ki > 100000 nM T47094 CYBO34 44266493 Ki > 100000 nM T47094 CQ18SV 44266551 Ki > 100000 nM T47094 C5Q9SI 44266599 Ki > 100000 nM T47094 CI0B2Z 44270410 IC50 = 22.3 nM T47094 CN95TJ 44270464 IC50 = 12.2 nM T47094 CHB1D5 44270481 IC50 = 32.7 nM T47094 C5EJ7N 44270504 IC50 = 1.3 nM T47094 C3QV8P 44270548 IC50 = 332 nM T47094 CN6GC1 44273822 IC50 = 3.3 nM T47094 C6ML4S 44274104 IC50 = 6.3 nM T47094 CR6B2W 44274118 IC50 = 5.6 nM T47094 CO31WA 44274153 IC50 = 0.27 nM T47094 C7KX6R 44274166 IC50 = 0.19 nM T47094 CQ06KN 44274167 IC50 = 14 nM T47094 C7IV8X 44274170 IC50 = 5.5 nM T47094 CW4GM5 44274180 IC50 = 0.79 nM T47094 CEZJ34 44274181 IC50 = 8.9 nM T47094 CFPX41 44274183 IC50 = 4.9 nM T47094 C2LQ4F 44274199 IC50 = 5.5 nM T47094 CUMX69 44274207 IC50 = 0.12 nM T47094 CVDQ61 44274242 IC50 = 570 nM T47094 CWH38F 44274251 IC50 = 0.14 nM T47094 CQY8F5 44274253 IC50 = 0.22 nM T47094 CEM8H6 44274254 IC50 = 950 nM T47094 CGU8T9 44274269 IC50 = 1.7 nM T47094 C4CA2F 44274277 IC50 = 2.3 nM T47094 CZ0H6C 44274316 IC50 = 15 nM T47094 CL9J8X 44274326 IC50 = 87 nM T47094 C1F6DO 44274331 IC50 = 8 nM T47094 CFG81H 44274341 IC50 = 31 nM T47094 C7A5XI 44274362 IC50 = 2.9 nM T47094 CGY2A0 44274392 IC50 = 82 nM T47094 C1CG0V 44274412 IC50 = 1.5 nM T47094 CH01FI 44274444 IC50 = 96 nM T47094 CS7IH8 44274520 IC50 = 42 nM T47094 C95YWC 44274530 IC50 = 5.2 nM T47094 C2OH7T 44274534 IC50 = 89 nM T47094 CK42GP 44274544 IC50 = 0.92 nM T47094 CGW01I 44274545 IC50 = 103 nM T47094 CTY6W2 44275987 IC50 = 33.3 nM T47094 CQ04LU 44276673 IC50 = 108 nM T47094 C5Q0GV 44276728 IC50 = 14 nM T47094 C5Y3BZ 44276732 IC50 = 34 nM T47094 C8YE9F 44276738 IC50 = 272 nM T47094 COV21W 44276788 IC50 = 7 nM T47094 CPC5E6 44276792 IC50 = 892 nM T47094 C4R9MX 44276856 IC50 >= 157 nM T47094 C2OJ9I 44276882 IC50 = 3.7 nM T47094 CG9JX6 44277452 IC50 = 48 nM T47094 CNP08Q 44277478 IC50 = 197 nM T47094 C2DA4T 44277705 IC50 = 288.4 nM T47094 C1GS4E 44277726 IC50 = 20.89 nM T47094 CSD41B 44277742 IC50 = 183 nM T47094 CM6CK5 44278425 IC50 = 2 nM T47094 C6XHU4 44278580 IC50 = 65 nM T47094 CT06IA 44281332 Ki = 100 nM T47094 CW6U9X 44281334 Ki = 115 nM T47094 C1K3ZC 44281345 Ki = 140 nM T47094 C2UL9J 44281357 Ki = 23 nM T47094 CUYH47 44281358 Ki = 92 nM T47094 C52GFN 44281392 Ki = 39 nM T47094 C7N0OI 44281476 Ki = 81 nM T47094 C0TB5X 44281505 Ki = 113 nM T47094 CA1I8S 44281516 Ki = 70 nM T47094 CTVS72 44281538 Ki = 10 nM T47094 CQ3W5Y 44281571 Ki = 5 nM T47094 C07XYA 44281572 Ki = 32 nM T47094 CH6UM7 44281587 Ki = 12 nM T47094 CXR0C9 44281633 Ki = 2 nM T47094 C1FK2S 44281649 Ki = 2 nM T47094 CL9IQ2 44281650 Ki = 2 nM T47094 C7S2TC 44281666 Ki = 2 nM T47094 C08YIH 44281672 Ki = 9 nM T47094 C9ZR1S 44281685 Ki = 10 nM T47094 CHV15K 44281713 Ki = 33 nM T47094 CQ92BL 44281743 Ki = 75 nM T47094 C4D1JN 44281744 Ki = 435 nM T47094 C6H5UG 44281753 Ki = 96 nM T47094 C5O9BF 44281769 IC50 = 9300 nM T47094 CME9G6 44281771 Ki = 53 nM T47094 C37KZY 44281776 Ki = 32 nM T47094 CS4D1T 44281778 Ki = 26 nM T47094 CO6YR1 44281784 Ki = 168 nM T47094 C4QZ8K 44281787 Ki = 58 nM T47094 C8AOU7 44281788 Ki = 33 nM T47094 CR2X6V 44281957 Ki = 6 nM T47094 C1S5QC 44281958 Ki = 7 nM T47094 CJ2SU9 44281976 Ki = 5 nM T47094 CZ58US 44281977 Ki = 1 nM T47094 C10-JUN 44282001 Ki = 5 nM T47094 C4O6IF 44282002 Ki = 13 nM T47094 CBE5C7 44282003 Ki = 42 nM T47094 C80LGR 44282004 Ki = 50 nM T47094 CWR82G 44286718 IC50 = 526 nM T47094 C6S4FR 44286754 IC50 = 593 nM T47094 CY9X5I 44286772 IC50 = 46 nM T47094 C3D7FC 44286798 IC50 = 297 nM T47094 CKA4Y3 44287191 IC50 = 56 nM T47094 C5TVJ4 44287210 IC50 = 235 nM T47094 C4T6WJ 44287211 IC50 = 121 nM T47094 C4Y0UD 44287368 IC50 = 301 nM T47094 CKY28E 44287388 IC50 = 323 nM T47094 C7P6MT 44287390 IC50 = 3917 nM T47094 CX39ER 44287409 IC50 = 3005 nM T47094 C5LMT4 44287443 IC50 = 51 nM T47094 C2PZW3 44287461 IC50 = 304 nM T47094 CE8U9V 44287481 IC50 = 620 nM T47094 CCD16S 44287503 IC50 = 112 nM T47094 C5W2OZ 44287511 IC50 = 47 nM T47094 C2G3DE 44287541 IC50 = 114 nM T47094 CKZP45 44287555 IC50 = 378 nM T47094 CIR8T1 44287556 IC50 = 45 nM T47094 CQSX53 44287557 IC50 = 226 nM T47094 CF8A0I 44287606 IC50 = 83 nM T47094 C83SQT 44287609 IC50 = 15 nM T47094 COX2E5 44287803 IC50 = 9 nM T47094 C2U5RV 44287861 IC50 = 370 nM T47094 CDNX43 44287895 IC50 = 38 nM T47094 CB59WY 44288548 IC50 = 19 nM T47094 C2VG8B 44288758 IC50 = 70 nM T47094 CEN36W 44288770 IC50 = 880 nM T47094 C3DWX6 44288772 IC50 = 210 nM T47094 CF8WO6 44288789 IC50 = 1380.38 nM T47094 C2NA3J 44288790 IC50 = 19 nM T47094 CY9Z4V 44288795 IC50 = 520 nM T47094 C3QHU8 44288846 IC50 = 110 nM T47094 C41HKF 44288885 IC50 = 12 nM T47094 CQ5V9I 44288892 IC50 = 220 nM T47094 CQC6I2 44288896 IC50 = 48 nM T47094 C1JH4R 44288901 IC50 = 11 nM T47094 CS90OI 44288926 IC50 = 24 nM T47094 CG32ZY 44288927 IC50 = 26 nM T47094 C83TZV 44288934 IC50 = 600 nM T47094 CPLM56 44288936 IC50 = 390 nM T47094 CLE4W1 44288951 IC50 = 20 nM T47094 C1CG2D 44288976 IC50 = 54 nM T47094 CNO4R2 44289102 IC50 = 92 nM T47094 CU4A3G 44289168 IC50 = 220 nM T47094 C3KJC1 44289169 IC50 = 130 nM T47094 C39SFB 44289191 IC50 > 10000 nM T47094 C31FPA 44289218 IC50 = 72 nM T47094 C8X2IA 44289219 IC50 = 60 nM T47094 C18OWF 44289232 IC50 = 1040 nM T47094 CR7NQ0 44289256 IC50 = 3300 nM T47094 CMG2P3 44289257 IC50 = 1380 nM T47094 CA2X9T 44289417 Ki < 100 nM T47094 C9X2VU 44289441 IC50 = 34 nM T47094 CMS30H 44289443 IC50 = 10.8 nM T47094 C48HJX 44289642 Ki < 100 nM T47094 CA0T2Z 44289862 IC50 = 3.3 nM T47094 C9J5PS 44289934 IC50 = 6 nM T47094 C3EM4V 44290030 IC50 = 8.3 nM T47094 CBV7T5 44290080 IC50 = 9.7 nM T47094 CFKB43 44291015 IC50 > 10000 nM T47094 CH16ID 44291515 IC50 = 10000 nM T47094 CEA5M3 44291788 IC50 = 10000 nM T47094 CC59NP 44294194 IC50 = 130 nM T47094 CLC2O3 44294224 IC50 = 2.4 nM T47094 C7OIV3 44294261 IC50 = 4.2 nM T47094 CI1U2D 44294291 IC50 = 0.62 nM T47094 COB7N8 44294293 IC50 = 0.2 nM T47094 CF52ZM 44294476 IC50 = 1400 nM T47094 CO37IY 44294481 IC50 = 22 nM T47094 CV80DA 44294519 IC50 = 2.1 nM T47094 C37OCJ 44294535 IC50 = 1.2 nM T47094 CLHM64 44294659 IC50 = 0.26 nM T47094 CK7E2B 44294660 IC50 = 0.42 nM T47094 CR2W3U 44294689 IC50 = 0.85 nM T47094 CT27IP 44295002 IC50 = 0.13 nM T47094 CF14MC 44297293 IC50 = 13 nM T47094 C0Q2XB 44297359 IC50 = 71 nM T47094 CMAB30 44297424 IC50 = 157 nM T47094 CJ8N9K 44297434 IC50 = 3.3 nM T47094 CA08QW 44297451 IC50 = 542 nM T47094 C6YJP9 44297463 IC50 = 60 nM T47094 C3HP1X 44297466 IC50 = 27 nM T47094 CX85ZL 44297469 IC50 = 58 nM T47094 C4D1BO 44297484 IC50 = 80 nM T47094 CJO19X 44297487 IC50 = 153 nM T47094 CI92PH 44297488 IC50 = 152 nM T47094 C92TCA 44297491 IC50 = 120 nM T47094 CCSD86 44297492 IC50 = 33 nM T47094 C0LG9U 44297493 IC50 = 57 nM T47094 CT53EF 44297498 IC50 = 36 nM T47094 CVA4E3 44297513 IC50 = 55 nM T47094 CIO68G 44297520 IC50 = 2000 nM T47094 CF27HC 44297523 IC50 = 88 nM T47094 C2L3RU 44297562 IC50 = 43 nM T47094 CH7BS2 44297563 IC50 = 260 nM T47094 CA65MF 44297602 IC50 = 54 nM T47094 CRD65Q 44297603 IC50 = 11 nM T47094 CKCI18 44297604 IC50 = 34 nM T47094 C0S5XL 44297605 IC50 = 1 nM T47094 C8KET4 44297629 IC50 = 7.7 nM T47094 CHZP06 44297642 IC50 = 6.6 nM T47094 CXL65U 44297648 IC50 = 24 nM T47094 CP01JD 44297649 IC50 = 63 nM T47094 C0BPQ7 44297680 IC50 = 18 nM T47094 C7HBL1 44297683 IC50 = 12 nM T47094 C8GWZ9 44297685 IC50 = 895 nM T47094 CX67HW 44297698 IC50 = 79 nM T47094 C57PHO 44297701 IC50 = 42 nM T47094 CS7JR3 44297705 IC50 = 163 nM T47094 C5KTA1 44297708 IC50 = 170 nM T47094 CC7ZF4 44297724 IC50 = 455 nM T47094 CS7IO9 44297728 IC50 = 1300 nM T47094 C8ADI4 44297749 IC50 = 100 nM T47094 CCYX86 44297753 IC50 = 263 nM T47094 CD9ZU5 44297822 IC50 = 382 nM T47094 C1E9OA 44297858 IC50 = 17 nM T47094 CC0O9R 44297859 IC50 = 61 nM T47094 C9TVE8 44297912 IC50 = 13 nM T47094 CT37HI 44297931 IC50 = 558 nM T47094 CL38HE 44297939 IC50 = 330 nM T47094 CA1VI9 44298065 IC50 = 2500 nM T47094 C1A5CW 44299271 IC50 = 0.5248 nM T47094 C9R7BI 44299273 IC50 = 2.2 nM T47094 CWT9J2 44299298 IC50 = 400 nM T47094 C6J5SQ 44299310 IC50 = 75 nM T47094 C79JTX 44299444 IC50 = 17 nM T47094 CAS17Q 44299463 IC50 = 9.7 nM T47094 C6WUX4 44299464 IC50 = 11.3 nM T47094 CBOM36 44299583 IC50 = 13.3 nM T47094 CUNI75 44299750 IC50 = 150 nM T47094 CZL24J 44299753 IC50 = 77 nM T47094 CER76I 44299814 IC50 = 2530 nM T47094 C0VO2P 44299829 IC50 = 1130 nM T47094 CR2WK9 44299830 IC50 = 87 nM T47094 C7C4IY 44299854 IC50 = 1530 nM T47094 C2V0HP 44299875 IC50 = 14 nM T47094 C4F1VL 44299876 IC50 = 82 nM T47094 C0B7FQ 44299898 IC50 = 93 nM T47094 CQ69CU 44299916 IC50 = 55 nM T47094 C9H2ED 44299943 IC50 = 6.8 nM T47094 CFJ3Z0 44299969 IC50 = 12.7 nM T47094 C6S7VY 44302017 IC50 = 430 nM T47094 CO43GA 44303835 IC50 = 280 nM T47094 C2SY0Z 44304123 IC50 = 3000 nM T47094 C0FUG2 44304301 Ki = 39.81 nM T47094 C2Y4FO 44304302 Ki = 1000 nM T47094 C3PU9W 44304323 Ki = 794.33 nM T47094 C98RBS 44304340 Ki = 316.23 nM T47094 C93EOA 44304381 Ki = 630.96 nM T47094 CVHI12 44304397 Ki = 1000 nM T47094 C9N2YP 44304398 Ki = 31.62 nM T47094 CY5R7N 44305221 IC50 = 0.7 nM T47094 C7WI6B 44305248 IC50 = 1 nM T47094 CPI9T3 44305271 IC50 = 4 nM T47094 C1LDB0 44305288 IC50 = 0.6 nM T47094 C3V1BM 44305467 IC50 = 3.5 nM T47094 C1UBW2 44305511 IC50 = 34 nM T47094 C97DBP 44305544 IC50 = 3 nM T47094 CCHD47 44305557 IC50 = 9 nM T47094 C5UTO0 44305711 IC50 > 1000 nM T47094 CQY7G9 44305817 Ki = 1.5 nM T47094 C04SCG 44305928 Ki = 2.4 nM T47094 CV2PA4 44307089 IC50 = 35 nM T47094 CW9HJ0 44307090 IC50 = 85 nM T47094 CDQ9M2 44307118 IC50 = 25 nM T47094 C62AMP 44307137 IC50 = 68 nM T47094 CQZ2B3 44307162 IC50 = 110 nM T47094 CO0Y3W 44307181 IC50 = 1.8 nM T47094 C7FZ5B 44307409 IC50 = 227 nM T47094 CAKQ84 44307416 IC50 = 0.63 nM T47094 CY4TG7 44307417 IC50 = 2.7 nM T47094 CHEC65 44308430 EC50 = 11 nM T47094 CRT79O 44308431 EC50 = 180 nM T47094 C6ONP4 44308550 EC50 = 5 nM T47094 CK8W5Q 44308551 EC50 > 10000 nM T47094 CY15MK 44308930 IC50 = 55 nM T47094 C8PB4F 44308931 IC50 = 2500 nM T47094 CRFO30 44312000 IC50 = 77 nM T47094 C05TAD 44312026 IC50 = 1033 nM T47094 C1W0GK 44312028 IC50 = 480 nM T47094 CX9PD5 44312056 IC50 = 10 nM T47094 CIA8X7 44312057 IC50 = 0.58 nM T47094 CX2LK5 44312145 IC50 = 332 nM T47094 C1LW7N 44312218 IC50 = 1100 nM T47094 C0B2IC 44312219 IC50 = 227 nM T47094 C5V9WG 44312256 IC50 = 23 nM T47094 C5G3YW 44312257 IC50 = 14 nM T47094 CI7NK6 44312285 IC50 = 1 nM T47094 CW0C3U 44312324 IC50 = 242 nM T47094 C7Q9IB 44313273 IC50 = 0.73 nM T47094 CRD1X4 44314154 Ki = 30 nM T47094 CFO10R 44314298 Ki = 62 nM T47094 CA78GB 44314299 Ki = 24 nM T47094 CO84ZW 44314453 Ki = 136 nM T47094 C4O8RX 44314454 Ki = 125 nM T47094 CJTI39 44314476 Ki = 33 nM T47094 CPH94L 44314480 Ki = 0.7 nM T47094 CX6Y2B 44314481 Ki = 34 nM T47094 CGY3S5 44314482 Ki = 25 nM T47094 CG9C8F 44314486 Ki = 14 nM T47094 CQ2IB5 44314487 Ki = 9 nM T47094 CYV8U9 44314502 Ki = 16 nM T47094 CQ5W1O 44314503 Ki = 22 nM T47094 CY59OC 44314504 Ki = 23 nM T47094 C43KGB 44314533 Ki = 82 nM T47094 CG7MS4 44314547 Ki = 181 nM T47094 CMX0D9 44314548 Ki = 70 nM T47094 CFK43V 44314577 Ki = 24 nM T47094 C5U8QB 44314578 Ki = 20 nM T47094 CHP4L1 44314597 Ki = 61 nM T47094 C10WAI 44314732 Ki = 136 nM T47094 CF12UM 44314834 Ki = 53 nM T47094 CF8EK6 44314861 Ki = 5 nM T47094 C87BVG 44314865 Ki = 113 nM T47094 CW4L2A 44314866 Ki = 125 nM T47094 CDX9O1 44314867 Ki = 4 nM T47094 C9VZE7 44314868 Ki = 9 nM T47094 CP0L4F 44314871 Ki = 19 nM T47094 CC7VT0 44314872 Ki = 47 nM T47094 CF2SA5 44314873 Ki = 13 nM T47094 CDHG71 44314945 Ki = 39 nM T47094 C4S3BF 44314946 Ki = 82 nM T47094 C3J6QU 44315209 Ki = 2.3 nM T47094 CH30NT 44315210 Ki = 2 nM T47094 C9PT3J 44315231 Ki = 2.7 nM T47094 CM9KT1 44315267 Ki = 157 nM T47094 CKT98C 44315297 Ki = 1.6 nM T47094 CAT8U5 44315298 Ki = 1.1 nM T47094 CF50BD 44315299 Ki = 2.4 nM T47094 CF2EQ0 44315369 Ki = 1.5 nM T47094 C70HNK 44315370 Ki = 1 nM T47094 C4GLI3 44315390 Ki = 1.3 nM T47094 C1S2MC 44315421 Ki = 1.2 nM T47094 CCW50R 44315422 Ki = 2.4 nM T47094 C46IEH 44315483 Ki = 0.6 nM T47094 C6TRV5 44315572 Ki = 2.5 nM T47094 CS9K4I 44315573 Ki = 3.2 nM T47094 CHX17S 44315576 Ki = 1.3 nM T47094 CDX84T 44315589 Ki = 1.9 nM T47094 C94WGI 44315590 Ki = 3 nM T47094 C0UK2L 44315591 Ki = 2.4 nM T47094 C24BAP 44318269 Ki = 245.47 nM T47094 CFI13C 44318310 IC50 = 513 nM T47094 C92EYC 44318312 Ki = 400 nM T47094 C9JCV8 44318349 IC50 = 183 nM T47094 CO3JG2 44318405 IC50 = 13 nM T47094 CFMC56 44318406 IC50 = 24 nM T47094 CR5CX6 44318413 IC50 = 30 nM T47094 CR06PH 44318455 Ki = 107.15 nM T47094 CV6ZX1 44318486 Ki = 74.13 nM T47094 C7G0DB 44318497 Ki = 457.09 nM T47094 C67YWG 44318565 Ki = 45.71 nM T47094 C5MOP3 44318578 Ki = 2041.74 nM T47094 CWE2I4 44318589 IC50 = 0.1 nM T47094 CHK73N 44318593 Ki = 575.44 nM T47094 COT68H 44318605 IC50 = 1.3 nM T47094 CJEB18 44318640 IC50 = 2.8 nM T47094 CSKF29 44318657 IC50 = 10 nM T47094 CC7X4U 44318658 IC50 = 16 nM T47094 CJSU01 44318665 Ki = 131.83 nM T47094 CX6G8W 44318671 IC50 = 99 nM T47094 CLN0J4 44318672 IC50 = 1.4 nM T47094 C42MUF 44318677 Ki = 1479.11 nM T47094 C5E8FK 44318685 IC50 = 1.1 nM T47094 CKE06V 44318694 Ki = 138.04 nM T47094 CQ6VO3 44318865 Ki = 1698.24 nM T47094 C47SWH 44318874 Ki = 645.65 nM T47094 C7Z2XQ 44319329 IC50 = 7 nM T47094 CQ9V1U 44319571 IC50 = 300 nM T47094 CB6H8C 44321046 IC50 = 67.61 nM T47094 CWD83P 44321047 IC50 = 487 nM T47094 C48PRB 44321049 IC50 > 32000 nM T47094 CJC4P6 44321099 IC50 = 383 nM T47094 C67LFG 44321408 IC50 = 16.6 nM T47094 CY6CB4 44321430 IC50 = 28000 nM T47094 C8MQ6N 44321442 IC50 = 19.95 nM T47094 CKC68E 44321456 IC50 = 16 nM T47094 CCLV78 44321457 IC50 = 1905.46 nM T47094 CKAI97 44321493 IC50 = 67.7 nM T47094 CK61BO 44321519 IC50 = 343 nM T47094 CU07XD 44322406 IC50 = 31.62 nM T47094 C0PN1I 44322429 IC50 = 199.53 nM T47094 CR5Z4U 44322511 IC50 = 316.23 nM T47094 C1MRC9 44322515 IC50 = 31.62 nM T47094 C32RKT 44322524 IC50 = 125.89 nM T47094 CJ3E6I 44322525 IC50 = 100 nM T47094 CLE8Z7 44322610 IC50 = 199.53 nM T47094 C3G0PJ 44322648 IC50 = 100 nM T47094 C2WYQ9 44322649 IC50 = 125.89 nM T47094 CF5KC1 44322678 IC50 = 1258.93 nM T47094 CQY03C 44322704 IC50 = 125.89 nM T47094 C60PEF 44322724 IC50 = 79.43 nM T47094 C29IOT 44322728 IC50 = 25.12 nM T47094 C4XEZ6 44322735 IC50 = 25.12 nM T47094 CFL9S1 44322736 IC50 = 50.12 nM T47094 CEI36U 44323563 Ki = 39.81 nM T47094 CR75NI 44324527 IC50 = 57 nM T47094 CG92NL 44324531 IC50 = 597 nM T47094 C2X4UJ 44324532 IC50 = 55 nM T47094 C2E8WF 44324681 IC50 = 930 nM T47094 CX2K9B 44324705 IC50 = 1080 nM T47094 C8H0VN 44324706 IC50 = 200 nM T47094 CPA57S 44324710 IC50 = 140 nM T47094 CY69DA 44324746 IC50 = 267 nM T47094 CC1U8F 44324775 IC50 = 9 nM T47094 CFH9Q5 44324793 IC50 = 9 nM T47094 CTK3J7 44324814 IC50 = 11 nM T47094 C9W4UZ 44324845 IC50 = 217 nM T47094 C25ZKE 44325035 IC50 = 0.89 nM T47094 CP5JO3 44325058 IC50 = 0.11 nM T47094 CKNZ89 44325096 IC50 = 6.5 nM T47094 C3B7PQ 44326280 IC50 = 13.7 nM T47094 CI8T3A 44326281 IC50 = 30 nM T47094 C6FR2K 44326290 IC50 = 135 nM T47094 CNE2L3 44326306 IC50 = 20 nM T47094 C2UD6S 44326328 IC50 = 49 nM T47094 C3WP5N 44326361 IC50 = 5.8 nM T47094 CBZ4Y8 44326362 IC50 = 4.3 nM T47094 CG0D6Q 44327794 IC50 = 10.87 nM T47094 CLHV50 44328357 IC50 = 4400 nM T47094 C6O0AR 44328374 IC50 = 1.9 nM T47094 C3K8CT 44328389 IC50 = 68 nM T47094 CXO21D 44328394 IC50 = 2.4 nM T47094 C72WYB 44328395 IC50 = 4800 nM T47094 C83CVT 44328400 IC50 = 7.1 nM T47094 C07CKN 44328401 IC50 = 170 nM T47094 C05ATS 44328405 IC50 = 39 nM T47094 CQ1V9A 44328407 IC50 = 230 nM T47094 CJD5R2 44328416 IC50 = 1100 nM T47094 C9G3CS 44328423 IC50 = 3.3 nM T47094 CI5U0A 44328424 IC50 = 7.2 nM T47094 CZQ5J6 44328425 IC50 = 4.1 nM T47094 CC09MS 44328454 IC50 = 0.14 nM T47094 C48ECR 44328469 IC50 = 0.92 nM T47094 CQ02YL 44328545 IC50 = 58 nM T47094 CF4MV5 44333527 IC50 > 10000 nM T47094 C91VWM 44333561 IC50 = 21 nM T47094 C82HEZ 44333579 IC50 = 100 nM T47094 C0B4UO 44333606 IC50 = 600 nM T47094 C74ECT 44333607 IC50 = 0.78 nM T47094 C4F8BK 44333682 IC50 = 52 nM T47094 C12WIP 44333692 IC50 = 1.3 nM T47094 C35ZCT 44333708 IC50 = 11 nM T47094 CNLI08 44333727 IC50 = 27 nM T47094 CNG70E 44333730 IC50 = 0.16 nM T47094 C73LIU 44333821 IC50 = 13 nM T47094 C7FY4N 44333950 IC50 = 14 nM T47094 CM3KT9 44333964 IC50 = 2.9 nM T47094 C3K7ST 44334006 IC50 = 55 nM T47094 CW5L3K 44334072 IC50 = 9 nM T47094 C1Z3FE 44334098 IC50 = 190 nM T47094 COQ67N 44334107 IC50 = 0.53 nM T47094 CMU3A1 44334108 IC50 = 2.2 nM T47094 C3I2WL 44334111 IC50 = 29 nM T47094 C70UVM 44334112 IC50 = 14 nM T47094 CZD2V6 44334113 IC50 = 30 nM T47094 CAPL13 44334114 IC50 = 0.13 nM T47094 CP6RO5 44334127 IC50 = 0.55 nM T47094 CUK2T6 44334143 IC50 = 13 nM T47094 CB2V8G 44334149 IC50 = 0.35 nM T47094 CWT5C2 44334185 IC50 = 2670 nM T47094 C38ELU 44334275 IC50 = 0.34 nM T47094 CCIH71 44334489 Ki = 512.86 nM T47094 CC9R7Z 44334499 Ki = 8.318 nM T47094 C9HA7L 44334500 Ki = 4265.8 nM T47094 C9V5LE 44334501 Ki = 1071.52 nM T47094 CVJZ64 44334581 Ki = 501.19 nM T47094 C2FNT4 44334582 Ki = 794.33 nM T47094 CFD3W6 44334591 Ki = 263.03 nM T47094 CN86UX 44334630 Ki = 75.86 nM T47094 CMN93Y 44334654 Ki = 38.9 nM T47094 C6DPW3 44334664 Ki = 2344.23 nM T47094 C9Y0HQ 44334665 Ki = 2290.87 nM T47094 CEOX43 44334666 Ki = 30.9 nM T47094 CGJ17C 44334708 Ki = 302 nM T47094 CU08PE 44334845 Ki = 30.2 nM T47094 CRMZ78 44335318 IC50 = 1 nM T47094 CQRG01 44335319 IC50 = 1.4 nM T47094 C38XWO 44335354 IC50 = 3.6 nM T47094 C9IB8V 44335360 IC50 = 6.4 nM T47094 CECZ64 44335372 IC50 = 1.1 nM T47094 CMF9U8 44335376 IC50 = 20 nM T47094 C3KP7V 44335410 IC50 = 12 nM T47094 CZKP39 44335466 IC50 = 18 nM T47094 C62MLD 44336987 Ki = 37 nM T47094 C5M2EF 44337007 Ki = 32 nM T47094 C70YEO 44337023 Ki = 28 nM T47094 C0S1MJ 44337024 Ki = 48 nM T47094 C2QUC4 44337078 Ki = 110 nM T47094 COC3Y7 44337079 Ki = 48 nM T47094 C79RVK 44337080 Ki = 148 nM T47094 C9KFY3 44337173 Ki = 92 nM T47094 CF0M7V 44337174 Ki = 15 nM T47094 CME07I 44337200 Ki = 13 nM T47094 C1I6ZY 44337201 Ki = 0.9 nM T47094 C24XSU 44337202 Ki = 48 nM T47094 C59BDG 44337207 Ki = 11 nM T47094 CG8RD6 44337208 Ki = 42 nM T47094 C8A1CW 44337266 Ki = 93 nM T47094 C1SUX0 44337270 Ki = 32 nM T47094 CWB0E3 44337288 Ki = 7.7 nM T47094 CY4XF2 44337289 Ki = 7.1 nM T47094 C9M2AX 44337308 Ki = 23 nM T47094 CE0XL3 44337313 Ki = 25 nM T47094 C1HLR5 44337324 Ki = 70 nM T47094 CNQS47 44337330 Ki = 21 nM T47094 CQ6B2X 44337353 Ki = 143 nM T47094 C3TM4J 44337354 Ki = 52 nM T47094 CI2TP9 44337355 Ki = 35 nM T47094 C8Z4UQ 44337370 Ki = 1.8 nM T47094 CKT4Z8 44337371 Ki = 3.2 nM T47094 C7NH1L 44337372 Ki > 1000 nM T47094 CA0QJ4 44337414 Ki = 30 nM T47094 C9EO0J 44337417 Ki > 1000 nM T47094 CR1G2S 44337421 IC50 = 3200 nM T47094 CWM3T9 44337428 IC50 = 1000 nM T47094 CU1X6H 44337467 Ki = 17 nM T47094 C52VXZ 44337500 IC50 = 29400 nM T47094 CA9S5B 44337514 Ki = 135 nM T47094 C3LM6I 44337569 IC50 = 820 nM T47094 C2K5ZU 44337667 IC50 = 410 nM T47094 CY69SK 44337795 IC50 = 140 nM T47094 CY9NA1 44338346 IC50 = 3.162 nM T47094 C71DZQ 44338359 Ki = 1.585 nM T47094 C7N2JZ 44338510 Ki = 79.43 nM T47094 CI4X6H 44338517 Ki = 1 nM T47094 CWZ3X8 44338518 Ki = 1.585 nM T47094 C7W3OB 44338530 Ki = 199.53 nM T47094 C0H5ZF 44338531 Ki = 100 nM T47094 CL7G8R 44338532 Ki = 25.12 nM T47094 C3F4RC 44338545 IC50 = 1.259 nM T47094 CX9WN6 44338546 Ki = 12.59 nM T47094 C1P9SM 44338557 Ki = 398.11 nM T47094 C8DB9O 44338583 Ki = 3.162 nM T47094 C8MUK3 44338584 IC50 = 5.012 nM T47094 CQ09VF 44338586 Ki = 6.31 nM T47094 CYMX71 44338587 IC50 = 3.162 nM T47094 CZ5F2V 44338618 Ki = 5.012 nM T47094 CYAU27 44338638 IC50 = 12.59 nM T47094 C98LQP 44338639 IC50 = 25.12 nM T47094 CMYH92 44338640 Ki = 7.943 nM T47094 C3HP7S 44338646 IC50 = 39.81 nM T47094 C61LBF 44338652 Ki = 50.12 nM T47094 CDN01U 44344195 IC50 = 640 nM T47094 CE8V0Q 44344209 IC50 = 2300 nM T47094 CCG75B 44344231 IC50 = 30 nM T47094 CR5TL4 44344435 IC50 = 1000 nM T47094 C2ICD8 44344994 IC50 > 10000 nM T47094 CV1K5F 44344995 IC50 = 270 nM T47094 CO43EP 44345010 IC50 = 380 nM T47094 CWT0Y2 44345147 IC50 = 620 nM T47094 C3GS0Z 44345148 IC50 = 15 nM T47094 CT28VL 44345155 IC50 > 10000 nM T47094 C94HJF 44345156 IC50 = 710 nM T47094 C6QB2E 44345938 IC50 = 9300 nM T47094 CZ57BY 44346149 IC50 = 1.995 nM T47094 C5Z1VX 44346159 IC50 = 30.2 nM T47094 C0FA2H 44346175 IC50 = 25.7 nM T47094 CCZ6R5 44346199 IC50 = 1400 nM T47094 CN5BV8 44346200 IC50 = 8128.31 nM T47094 C67PJR 44346206 Ki = 1 nM T47094 CVAI62 44346234 IC50 = 0.3631 nM T47094 C1UC4P 44346259 IC50 = 1467 nM T47094 C3H0YL 44346302 IC50 = 128.82 nM T47094 CKWE64 44346319 IC50 = 1584.89 nM T47094 CYE29O 44346320 IC50 = 19.95 nM T47094 CP0KT1 44346330 IC50 = 1995.26 nM T47094 CO8SZ0 44346333 IC50 = 1258.93 nM T47094 CBX1T0 44346334 IC50 = 12.59 nM T47094 CPS56R 44346399 IC50 = 125.89 nM T47094 C3DR7K 44346420 IC50 = 22.91 nM T47094 CODT92 44346438 IC50 = 0.3981 nM T47094 C6TQ4L 44346476 IC50 = 2344.23 nM T47094 CJ7G0K 44346480 IC50 = 363.08 nM T47094 CL84VN 44346497 IC50 = 75.86 nM T47094 CT3UM5 44346524 IC50 = 229.09 nM T47094 CIF2M0 44346536 IC50 = 9.12 nM T47094 C98IJU 44346550 IC50 = 2344.23 nM T47094 CR5K6N 44346551 IC50 = 1.995 nM T47094 CGFI29 44346557 IC50 = 316.23 nM T47094 CV7G8P 44346558 IC50 = 5.012 nM T47094 CRZ5Y6 44346650 Ki > 10000 nM T47094 C7NC0K 44346664 IC50 = 2691.53 nM T47094 CQJX45 44346675 IC50 = 6025.6 nM T47094 CD6MW1 44346693 IC50 = 81.28 nM T47094 C9PM8F 44346694 IC50 = 10.72 nM T47094 CF91YC 44349303 IC50 = 54000 nM T47094 C5M7OK 44349304 IC50 = 26000 nM T47094 CFV0C3 44349310 IC50 > 100000 nM T47094 CLP9F2 44349349 IC50 > 100000 nM T47094 CH7U0I 44349364 IC50 = 38000 nM T47094 C3T4NY 44349369 IC50 = 98000 nM T47094 CQ5R8W 44349370 IC50 = 48000 nM T47094 CFZM03 44349375 IC50 = 88000 nM T47094 CHM95S 44349376 IC50 > 100000 nM T47094 CDL23P 44352062 IC50 = 340 nM T47094 C73TMR 44356378 IC50 = 0.19 nM T47094 C5D7ZO 44356404 IC50 = 0.29 nM T47094 CIHU84 44357006 IC50 = 0.19 nM T47094 C10RQO 44358247 Ki = 7.943 nM T47094 CZ1VH4 44358248 Ki = 31.62 nM T47094 CH27KL 44358249 Ki = 1.585 nM T47094 CUSY73 44358280 Ki = 3.162 nM T47094 CYF98W 44358317 Ki = 2.512 nM T47094 C98CJF 44358318 Ki = 1.995 nM T47094 C8P3DH 44358323 Ki = 3.162 nM T47094 C0IHV6 44358334 Ki = 3.162 nM T47094 C2MG1Q 44358335 Ki = 1.259 nM T47094 CRB94A 44358346 Ki = 100 nM T47094 CH2IP8 44358385 Ki = 251.19 nM T47094 C9LX8J 44358408 Ki = 15.85 nM T47094 C40EJQ 44358409 Ki = 19.95 nM T47094 C49CXZ 44358413 Ki = 63.1 nM T47094 CKMU12 44358416 IC50 = 210 nM T47094 CK14SR 44358421 Ki = 158.49 nM T47094 CTI27O 44358425 Ki = 2.512 nM T47094 CKTG19 44358426 IC50 = 3700 nM T47094 CV1EF0 44358427 IC50 = 6.4 nM T47094 CCY14W 44358428 IC50 = 1.4 nM T47094 C5C0HR 44358435 IC50 = 140 nM T47094 C7U9TR 44358442 IC50 = 32 nM T47094 C47ISC 44358456 Ki = 1.995 nM T47094 CGVM40 44358467 IC50 = 2.4 nM T47094 C6MPT3 44358469 IC50 = 5.2 nM T47094 CQ8GX6 44358470 IC50 = 1.7 nM T47094 CACM71 44358471 IC50 = 1.6 nM T47094 CT50QI 44358472 IC50 = 110 nM T47094 CFMG60 44358473 IC50 = 1500 nM T47094 CZF8M2 44358475 IC50 = 8.9 nM T47094 C1EBP2 44358476 IC50 = 7.6 nM T47094 CAFK20 44358495 IC50 = 2 nM T47094 CJK15Y 44358500 IC50 = 37 nM T47094 C3CUW5 44358516 Ki = 1 nM T47094 C8GLS5 44358519 IC50 = 5 nM T47094 CU4V2D 44358520 IC50 = 81 nM T47094 C8AY6D 44358545 IC50 = 5.4 nM T47094 CTR8U0 44358551 Ki = 63.1 nM T47094 CKAW07 44358552 IC50 = 22 nM T47094 C2D7XE 44358561 IC50 = 1.7 nM T47094 CCRB38 44358568 Ki = 10 nM T47094 C6Z9KO 44358569 Ki = 3.162 nM T47094 CZR75C 44358585 IC50 = 10 nM T47094 CFW25R 44358589 Ki = 125.89 nM T47094 CQ9DN1 44358596 IC50 = 14 nM T47094 C01DKJ 44358597 Ki = 15.85 nM T47094 C0L2TE 44358602 IC50 = 14 nM T47094 C2EB0M 44358603 IC50 = 1.1 nM T47094 CV94TU 44358604 IC50 = 1.4 nM T47094 CV2R3D 44358610 IC50 = 0.88 nM T47094 C9A8FQ 44358611 IC50 = 130 nM T47094 CFH61O 44358612 Ki = 1.585 nM T47094 CU07PC 44358649 IC50 = 130 nM T47094 CI2U4B 44358657 IC50 = 1.8 nM T47094 CIF46D 44358670 IC50 = 6.9 nM T47094 CR87LN 44358672 IC50 = 6 nM T47094 CD1CM5 44358673 IC50 = 130 nM T47094 CN59YM 44358676 IC50 = 1.3 nM T47094 CA1U6L 44358679 IC50 = 12 nM T47094 CDM0P9 44358680 IC50 = 12 nM T47094 CINP90 44358683 IC50 = 12 nM T47094 C0C7TW 44358703 IC50 = 4.3 nM T47094 C28FJT 44358707 IC50 = 1.5 nM T47094 CS17UD 44358708 IC50 = 15 nM T47094 CG4SK1 44358709 IC50 = 12 nM T47094 CK0DG5 44358710 IC50 = 16 nM T47094 C3IUH2 44358719 IC50 = 3 nM T47094 CV91OY 44358720 IC50 = 1.8 nM T47094 C8BO2S 44358727 IC50 = 2.1 nM T47094 CU41OC 44358731 IC50 = 0.75 nM T47094 C2QEU0 44358732 IC50 = 1.4 nM T47094 CI56QG 44358741 IC50 = 2.9 nM T47094 C96JNS 44358742 IC50 = 3 nM T47094 CM1C2O 44358767 IC50 = 2.9 nM T47094 CTX5A7 44358783 IC50 = 18.2 nM T47094 C8S4YT 44358801 IC50 = 151.36 nM T47094 CJ6QW8 44358814 IC50 = 34.67 nM T47094 C1S2GP 44358834 IC50 = 141.25 nM T47094 CO1V9W 44358847 IC50 = 97.72 nM T47094 CY3EQ4 44358861 IC50 = 42.66 nM T47094 CW92CG 44358864 IC50 = 4.8 nM T47094 C5CSR7 44358981 IC50 = 1584.89 nM T47094 CF7BO1 44358982 IC50 = 7244.36 nM T47094 CX25NJ 44359010 IC50 = 7413.1 nM T47094 CGE83J 44359025 IC50 = 15.85 nM T47094 C27ARD 44359054 IC50 = 2089.3 nM T47094 CS1L7U 44359055 IC50 = 3715.35 nM T47094 CX72YD 44359056 IC50 = 1096.48 nM T47094 CO40JL 44359071 IC50 = 2.138 nM T47094 CQFZ81 44359083 IC50 = 3.162 nM T47094 CNI6Z0 44359088 IC50 = 19.05 nM T47094 CM9BX3 44359091 IC50 = 10 nM T47094 CG2BC4 44359094 IC50 = 2.399 nM T47094 CA8PR6 44359096 IC50 = 22.39 nM T47094 C4BA2O 44359109 IC50 = 26.92 nM T47094 C6W1SE 44359111 IC50 = 19.95 nM T47094 C16AIL 44359117 IC50 = 12.88 nM T47094 CC73QO 44359259 IC50 = 33.11 nM T47094 C5UK8T 44359260 IC50 = 28.84 nM T47094 CV1G3I 44362586 IC50 = 107 nM T47094 CN9M7Q 44362598 IC50 = 103 nM T47094 CPK1M0 44363435 Ki = 69 nM T47094 C9JX1F 44363436 Ki = 20 nM T47094 C36NEP 44363442 Ki = 14 nM T47094 C5BGV8 44363756 Ki = 18 nM T47094 CL03EB 44363877 Ki = 44 nM T47094 C4P7HE 44363908 Ki = 18 nM T47094 CLT92R 44363909 Ki = 117 nM T47094 C97AKV 44363912 Ki = 36 nM T47094 C3SJ2T 44363925 Ki = 19 nM T47094 C7W8HN 44363926 Ki = 4 nM T47094 CUS74Z 44363936 Ki = 17 nM T47094 CXOL74 44363948 Ki = 36 nM T47094 C98HSV 44363949 Ki = 16 nM T47094 C5MKE6 44363952 Ki = 13 nM T47094 C4FMW7 44363962 Ki = 16 nM T47094 CO96ZG 44363963 Ki = 25 nM T47094 CN5Z4T 44363978 Ki = 38 nM T47094 C10SMA 44363979 Ki = 20 nM T47094 CM3E7F 44363982 Ki = 14 nM T47094 C8RFG9 44363983 Ki = 7 nM T47094 C0AF2Z 44363984 Ki = 13 nM T47094 C2W8KH 44363990 Ki = 14 nM T47094 CG5H8R 44364001 Ki = 112 nM T47094 C5UK4I 44364002 Ki = 8 nM T47094 CK91IA 44364003 Ki = 6 nM T47094 CY5O2B 44364030 Ki = 50 nM T47094 C0X1AS 44368082 IC50 = 15 nM T47094 C4CY9F 44368083 IC50 = 10 nM T47094 CI3XV1 44368118 IC50 = 13 nM T47094 C3DXC0 44368158 IC50 = 16 nM T47094 CU12YK 44368159 IC50 = 70 nM T47094 CSJ4K5 44368171 IC50 = 1.4 nM T47094 C7D9AK 44368172 IC50 = 5 nM T47094 CYH20X 44370340 IC50 = 3.5 nM T47094 CX7H8J 44370352 IC50 = 73 nM T47094 CRF46Y 44370354 IC50 = 1.8 nM T47094 C7YKA0 44370369 IC50 = 20 nM T47094 CMK71Z 44370448 IC50 = 1.4 nM T47094 CG3QL2 44370449 IC50 = 3.8 nM T47094 C9T2SB 44370769 IC50 = 33 nM T47094 CZ6Y3W 44370893 IC50 = 13 nM T47094 C9QKW7 44370925 IC50 = 8 nM T47094 CS25TE 44370928 IC50 = 5.5 nM T47094 CO1T4S 44370954 IC50 = 250 nM T47094 C4KY3R 44370973 IC50 = 1.8 nM T47094 CBI0T1 44375286 IC50 > 50000 nM T47094 CHW86C 44375297 IC50 ~ 50000 nM T47094 C9ZD6T 44375692 IC50 > 100000 nM T47094 C87PLB 44380062 Ki = 1 nM T47094 CH7UK2 44380069 Ki = 7.4 nM T47094 CK95JD 44380072 Ki = 0.4 nM T47094 CUP91D 44380079 Ki = 1.8 nM T47094 C41ZOW 44380081 Ki = 0.5 nM T47094 CO61AX 44380082 Ki = 0.7 nM T47094 C3Y1FS 44380090 Ki = 2.4 nM T47094 C81BCL 44380091 Ki = 0.7 nM T47094 CAM4W5 44380092 Ki = 1.9 nM T47094 CKFH38 44380093 Ki = 24 nM T47094 CUD8V6 44380094 Ki = 17 nM T47094 CP1N5F 44380095 Ki = 15 nM T47094 CUG0H7 44380107 Ki = 103 nM T47094 COCK40 44380131 Ki = 0.9 nM T47094 CZ4OK3 44380132 Ki = 0.8 nM T47094 CPC91W 44380206 Ki = 0.8 nM T47094 C3LA4N 44380248 Ki = 2.8 nM T47094 CV0S3A 44380249 Ki = 2.2 nM T47094 CW1RF0 44380277 Ki = 100 nM T47094 CDJ1I5 44380279 Ki = 1.2 nM T47094 C7SU4I 44380289 Ki = 1.7 nM T47094 CS30MR 44380290 Ki = 0.8 nM T47094 CAO4I2 44380313 Ki = 15 nM T47094 CGT8P4 44380337 Ki = 0.7 nM T47094 C5YBD1 44380338 Ki = 1.6 nM T47094 C4IE0V 44380396 Ki = 0.7 nM T47094 C93AGV 44380413 Ki = 2.2 nM T47094 CH0QX3 44380414 Ki = 1.2 nM T47094 CKR3J9 44380415 Ki = 0.9 nM T47094 C0BO2Q 44380448 Ki = 0.6 nM T47094 C0CN7P 44380457 Ki = 4.7 nM T47094 CI4GR9 44380473 Ki = 0.7 nM T47094 CJW1X3 44380474 Ki = 25 nM T47094 CN09IU 44380475 Ki = 33 nM T47094 C2SA3D 44380526 Ki = 1.5 nM T47094 CM7X5R 44380527 Ki = 17 nM T47094 CZ0O9E 44380596 Ki = 49 nM T47094 COJN63 44380680 Ki = 57 nM T47094 C2E5UX 44380707 IC50 = 160 nM T47094 CP6CN5 44380708 IC50 = 20 nM T47094 CM9PY4 44380709 IC50 = 700 nM T47094 C7LK2B 44380732 Ki = 20 nM T47094 C2WDA0 44380733 Ki = 7 nM T47094 CIKQ65 44380745 IC50 = 350 nM T47094 CHK0I5 44380763 Ki = 81 nM T47094 CO09YI 44380764 Ki = 38 nM T47094 CW30XT 44380794 Ki = 8 nM T47094 C9Z1VX 44380795 Ki = 25 nM T47094 C4RB9H 44381056 IC50 = 140 nM T47094 C3XM5O 44381059 IC50 = 240 nM T47094 C8KUZ9 44383265 IC50 = 86.3 nM T47094 C38UDJ 44383681 IC50 = 560 nM T47094 C4M0VW 44383815 IC50 = 310 nM T47094 CO24LE 44383969 IC50 = 53 nM T47094 CNKR49 44384677 IC50 = 65.9 nM T47094 C2JK9W 44384678 IC50 = 252 nM T47094 CX0N1K 44384901 IC50 = 634 nM T47094 CY43OG 44384902 IC50 = 107 nM T47094 CPRI69 44384986 IC50 = 64.1 nM T47094 C29NBY 44384987 IC50 = 69.9 nM T47094 CT8OC5 44385121 IC50 = 767 nM T47094 CD34IL 44385575 IC50 = 66.2 nM T47094 C2CI6G 44386105 IC50 = 138 nM T47094 C0V6SU 44386230 IC50 = 313 nM T47094 CR43OB 44386231 IC50 = 168 nM T47094 CR10NQ 44396809 IC50 = 12 nM T47094 CPX85J 44396853 IC50 = 1.6 nM T47094 CI6O9K 44402934 IC50 = 10 nM T47094 CX6V9Q 44404006 IC50 = 161 nM T47094 CH7Z3D 44407321 IC50 = 1 nM T47094 CFU2S7 44407325 IC50 = 0.13 nM T47094 CE2R3O 44407331 IC50 = 0.09 nM T47094 CHO57T 44407370 IC50 = 0.24 nM T47094 CS21QZ 44407422 IC50 = 1.2 nM T47094 CLG2U0 44407427 IC50 = 0.1 nM T47094 CUTS73 44407431 IC50 = 0.65 nM T47094 CCQX09 44407459 IC50 = 0.27 nM T47094 C9B4AK 44407467 IC50 = 2.1 nM T47094 CDPQ01 44407513 IC50 = 0.11 nM T47094 C0FT4M 44407890 Ki = 41 nM T47094 C24XHZ 44407896 Ki = 93 nM T47094 CE58BK 44407901 Ki = 19.95 nM T47094 CY3F0H 44407902 Ki = 1.585 nM T47094 CH1NT3 44407903 Ki = 6.31 nM T47094 CP6KU4 44407906 Ki = 6.31 nM T47094 CL2UO4 44407907 Ki = 10 nM T47094 CNGL40 44407908 Ki = 2.512 nM T47094 CQ05IJ 44407917 Ki = 10 nM T47094 C3D5OB 44407932 Ki = 89 nM T47094 CAF26T 44407938 Ki = 0.5 nM T47094 C1UEV0 44407939 Ki = 1.7 nM T47094 CAI9R6 44407971 Ki = 1.259 nM T47094 C7RX9A 44407972 Ki = 3.162 nM T47094 CQ53KC 44407998 Ki = 1.259 nM T47094 CKT09U 44408025 Ki = 0.3981 nM T47094 C8X6VN 44408033 Ki = 3.981 nM T47094 C15SZO 44408039 Ki = 0.7943 nM T47094 CNT06M 44408040 Ki = 2.512 nM T47094 CFZ2O7 44408045 Ki = 1.995 nM T47094 C9GHN1 44408046 Ki = 1.259 nM T47094 CFD63S 44408047 Ki = 0.7943 nM T47094 CRFS45 44408048 Ki = 6.31 nM T47094 C5SN6C 44408051 Ki = 12.59 nM T47094 COG01F 44408062 Ki = 2.7 nM T47094 CZF3W7 44408088 Ki = 10 nM T47094 C8IU4G 44408089 Ki = 12.59 nM T47094 CY1P0W 44408100 Ki = 3.1 nM T47094 C4J5SO 44408107 Ki = 0.8 nM T47094 CRB41P 44408123 IC50 = 0.8 nM T47094 CQPK26 44408124 IC50 = 1.1 nM T47094 C92YHJ 44408144 IC50 = 6.2 nM T47094 C35UHG 44408158 IC50 = 0.62 nM T47094 CF05TZ 44408176 IC50 = 0.5 nM T47094 CA94TU 44408177 IC50 = 0.48 nM T47094 CK4IB0 44408290 IC50 = 0.48 nM T47094 CDK7W3 44408291 IC50 = 0.48 nM T47094 CTM53U 44408295 IC50 = 1.5 nM T47094 CJE43Y 44408313 IC50 = 0.66 nM T47094 CQG14C 44408625 Ki = 295 nM T47094 CX83CN 44408628 Ki = 372 nM T47094 CH7Q6U 44408736 Ki = 22 nM T47094 CU21GY 44408755 Ki = 4 nM T47094 CMKF16 44408766 Ki = 3.8 nM T47094 C49QLZ 44408793 Ki > 10000 nM T47094 CV7XQ1 44408821 Ki = 68 nM T47094 CTQC73 44408838 Ki = 1.7 nM T47094 CP13XT 44408846 Ki = 6.2 nM T47094 CAP80G 44408864 Ki = 1380 nM T47094 C6IV9Z 44409000 Ki = 724 nM T47094 CP4I9L 44409004 Ki = 45 nM T47094 C8TX1R 44409008 Ki = 3.5 nM T47094 C5NZE8 44409023 Ki = 2 nM T47094 CP10EK 44410155 IC50 = 2.8 nM T47094 C9J0RV 44410162 IC50 = 4.2 nM T47094 C3YC0E 44410191 IC50 = 0.6 nM T47094 C5I4SO 44410193 IC50 = 1 nM T47094 CY69JU 44410194 IC50 = 9 nM T47094 CVB31D 44410278 IC50 = 0.5 nM T47094 CKWZ76 44410281 IC50 = 1.2 nM T47094 CQ8T0X 44410283 IC50 = 1.5 nM T47094 CYT96G 44410317 IC50 = 0.4 nM T47094 CWHE83 44410321 IC50 = 200 nM T47094 CGZ2J9 44411637 IC50 = 640 nM T47094 CE45QC 44411742 IC50 = 1000 nM T47094 CUB0V6 44412159 IC50 = 0.53 nM T47094 CO82EW 44412173 IC50 = 0.28 nM T47094 CACE19 44412207 IC50 = 0.14 nM T47094 CV4KZ7 44412225 IC50 = 0.64 nM T47094 CHF80Z 44412226 IC50 = 0.12 nM T47094 CCD01F 44412235 IC50 = 0.43 nM T47094 CECW41 44412236 IC50 = 0.19 nM T47094 C1D7YV 44412245 IC50 = 0.22 nM T47094 CH04GP 44412373 IC50 = 0.44 nM T47094 CYK1I6 44412374 IC50 = 0.33 nM T47094 CK5O6Q 44412445 IC50 = 0.23 nM T47094 CW71MS 44412453 IC50 = 0.49 nM T47094 C6R2ID 44412493 IC50 = 0.41 nM T47094 C2FRX1 44413144 IC50 = 650 nM T47094 C60KVA 44415392 IC50 = 2.4 nM T47094 C6MOZ8 44415393 IC50 = 260 nM T47094 C4DRF0 44415399 IC50 = 8.2 nM T47094 CI7XW0 44415400 IC50 = 0.89 nM T47094 C7UX1M 44415403 IC50 = 1.5 nM T47094 CDB1I7 44415404 IC50 = 0.81 nM T47094 C6T7RA 44415411 IC50 = 6.2 nM T47094 C62RHI 44415412 IC50 = 5.3 nM T47094 CNH80D 44415415 IC50 = 1.1 nM T47094 CAD36E 44415423 IC50 = 67 nM T47094 C95GWC 44415424 IC50 = 40 nM T47094 C9D1WP 44415435 IC50 = 7.2 nM T47094 CT32NY 44415436 IC50 = 2.7 nM T47094 CX17VO 44415437 IC50 = 300 nM T47094 C3F4KE 44415443 IC50 = 1.9 nM T47094 C9YLK5 44415444 IC50 = 0.77 nM T47094 CLQX71 44415447 IC50 = 7.9 nM T47094 CJLX19 44415448 IC50 = 2.7 nM T47094 C1BWV0 44415449 IC50 = 8.3 nM T47094 CCJM58 44415458 IC50 = 5 nM T47094 CGZ4N3 44415469 IC50 = 7.2 nM T47094 CQW1K5 44415470 IC50 = 100 nM T47094 C9R7VQ 44415471 IC50 = 2.1 nM T47094 CHT8F9 44415472 IC50 = 45 nM T47094 C1TX9P 44415484 IC50 = 2.3 nM T47094 CG07XA 44415485 IC50 = 1.9 nM T47094 CS1P2H 44415486 IC50 = 5.2 nM T47094 CRAV19 44415502 IC50 = 1.9 nM T47094 C2AGC6 44415513 IC50 = 3.5 nM T47094 C1U9RB 44415529 IC50 = 9.8 nM T47094 CJP49C 44415530 IC50 = 2.7 nM T47094 CA09WU 44415539 IC50 = 5 nM T47094 CP9Y7F 44415540 IC50 = 16 nM T47094 C0XSC4 44415550 IC50 = 0.83 nM T47094 CYTQ91 44415554 IC50 = 0.55 nM T47094 C5OQB8 44415789 IC50 = 0.28 nM T47094 CS5T0X 44415808 IC50 = 0.43 nM T47094 C90FIM 44415840 IC50 = 0.95 nM T47094 C8J3PY 44415869 IC50 = 0.25 nM T47094 CQM7T1 44415896 IC50 = 0.52 nM T47094 CL9Z3N 44415909 IC50 = 0.41 nM T47094 CXAD78 44415921 IC50 = 0.4 nM T47094 CKSJ35 44415947 IC50 = 0.6 nM T47094 CBDA42 44415967 IC50 = 0.7 nM T47094 CS2PB0 44415986 IC50 = 1.4 nM T47094 C4JKR8 44416008 IC50 = 0.27 nM T47094 CN0D8J 44416078 IC50 = 0.16 nM T47094 CAL45M 44416136 IC50 = 0.68 nM T47094 C25USR 44433393 IC50 = 0.6 nM T47094 CQC0U9 44433394 IC50 = 0.2 nM T47094 C93YCH 44433781 IC50 = 450 nM T47094 C2XPG0 44433782 IC50 = 142 nM T47094 C0NK9X 44433783 IC50 = 11 nM T47094 CO4VC6 44433784 IC50 = 0.68 nM T47094 CU2P9D 44433785 IC50 = 62 nM T47094 CI2Q6J 44433786 IC50 = 13 nM T47094 C3HMD2 44433787 IC50 = 0.79 nM T47094 C0RB1Y 44433788 IC50 = 4.1 nM T47094 C9LM7U 44433789 IC50 = 0.12 nM T47094 CFD93S 44433790 IC50 = 3.7 nM T47094 C28SOB 44433792 IC50 = 0.84 nM T47094 CA43ZS 44433793 IC50 = 0.74 nM T47094 CF4P6R 44433794 IC50 = 3.4 nM T47094 C5I9OY 44433795 IC50 = 24 nM T47094 CO71QT 44433796 IC50 = 0.58 nM T47094 CWDJ93 44433797 IC50 = 0.05 nM T47094 CU67NA 44433798 IC50 = 0.05 nM T47094 CNU4B6 44433799 IC50 = 8 nM T47094 C5V7WE 44433800 IC50 = 0.07 nM T47094 CBP25Q 44433802 IC50 = 0.17 nM T47094 CB1SD9 44433803 IC50 = 0.07 nM T47094 C50DTF 44433804 IC50 = 0.03 nM T47094 C95CMW 44433810 IC50 = 0.97 nM T47094 CC9U2N 44444629 IC50 = 0.24 nM T47094 CH2O6A 44444631 IC50 = 0.09 nM T47094 CA6XC8 44444634 IC50 = 0.07 nM T47094 C86XMD 44444637 IC50 = 0.09 nM T47094 C64SGU 44444638 IC50 = 0.15 nM T47094 CIAF97 44444640 IC50 = 0.18 nM T47094 CS3J1X 44444643 IC50 = 0.07 nM T47094 CQ72MI 44444646 IC50 = 0.12 nM T47094 CV1EH3 44444650 IC50 = 0.12 nM T47094 C2DCI5 44444654 IC50 = 0.34 nM T47094 CRJ94Z 44444658 IC50 = 0.11 nM T47094 C8AM7U 44444659 IC50 = 0.38 nM T47094 CIAZ93 44444660 IC50 = 0.16 nM T47094 C9D8YK 44444664 IC50 = 0.1 nM T47094 C5JN6M 44444666 IC50 = 0.06 nM T47094 CODZ34 44444669 IC50 = 0.14 nM T47094 CAP48O 44444671 IC50 = 0.3 nM T47094 CD4LE0 44444674 IC50 = 0.47 nM T47094 CVA47J 44444677 IC50 = 0.58 nM T47094 C1H7YR 44444681 IC50 = 0.11 nM T47094 C2YM7W 44444684 IC50 = 0.13 nM T47094 CK4VG2 44444685 IC50 = 0.09 nM T47094 CS07OF 44444688 IC50 = 0.11 nM T47094 C2DV4I 44444692 IC50 = 0.16 nM T47094 C7M6XU 44444693 IC50 = 0.12 nM T47094 CR78TC 44444694 IC50 = 0.18 nM T47094 CMG35V 44444695 IC50 = 0.13 nM T47094 C35RAO 44456522 IC50 = 0.14 nM T47094 C5SVZ4 44456524 IC50 = 0.27 nM T47094 CGL96P 44456580 IC50 = 1 nM T47094 CQD9F8 44456625 IC50 = 1.5 nM T47094 CDR6X5 44456650 IC50 = 1.2 nM T47094 C61GLN 44456651 IC50 = 3.6 nM T47094 C71NZI 44456700 IC50 = 0.28 nM T47094 C2WC6N 44456703 IC50 = 0.63 nM T47094 CGFB95 44456748 IC50 = 4.4 nM T47094 CN41BU 44456802 IC50 = 0.06 nM T47094 CLZ38B 44456828 IC50 = 0.88 nM T47094 CUJT56 44456847 IC50 = 2.7 nM T47094 C4HYX0 44456865 IC50 = 0.33 nM T47094 CT7V6D 44456866 IC50 = 7.8 nM T47094 C59WAV 44456894 IC50 = 1.3 nM T47094 CZE71N 44458328 IC50 = 1 nM T47094 C3X5CH 44458351 IC50 = 197 nM T47094 C7MC0Z 44458353 IC50 = 292 nM T47094 CPMZ84 44458598 IC50 = 8 nM T47094 CX0TU1 44458983 IC50 = 197 nM T47094 C0GUN2 44459032 IC50 = 30 nM T47094 CXF67K 44462338 Ki = 28 nM T47094 CG1QT9 44550460 Ki = 70.9 nM T47094 CS5LC7 44560754 Ki = 2 nM T47094 CKSW70 44560755 Ki = 0.9 nM T47094 CP27CT 44560773 Ki = 0.6 nM T47094 CT5K7N 44560774 Ki = 2.6 nM T47094 CCXS29 44560775 Ki = 0.3 nM T47094 CQ35IZ 44560809 Ki = 0.5 nM T47094 CSJ9U6 44560810 Ki = 0.2 nM T47094 C7FC3Q 44560811 Ki = 0.2 nM T47094 CL21VC 44560832 Ki = 0.4 nM T47094 C83GOJ 44560833 Ki = 0.5 nM T47094 CLMN13 44560834 Ki = 0.4 nM T47094 CRZ0I9 44575660 Ki = 170000 nM T47094 C3NKY2 44577989 IC50 = 0.4 nM T47094 C56MVE 44578023 IC50 < 0.1 nM T47094 CO7SW4 44578024 IC50 = 0.7 nM T47094 CF2T6X 44578025 IC50 < 0.1 nM T47094 CTB4E2 44578056 IC50 = 0.9 nM T47094 CF71YM 44578057 IC50 < 0.1 nM T47094 C9UJN1 44578095 IC50 < 0.1 nM T47094 CAWE52 44593632 IC50 < 0.1 nM T47094 CP37YX 44593633 IC50 = 0.4 nM T47094 CB8LX4 44593634 IC50 < 0.1 nM T47094 C29QEV 44593636 IC50 < 0.1 nM T47094 CD38TX 45259221 Ki = 1 nM T47094 C6MT0H 45259223 Ki = 1.995 nM T47094 CG8ZA5 45259228 Ki = 0.05012 nM T47094 CW1AP8 45259231 Ki = 0.03981 nM T47094 CPM39I 45263832 Ki = 0.05012 nM T47094 C6FEH0 45271306 Ki = 0.052 nM T47094 CV13DA 46224897 Ki = 50.12 nM T47094 CVM20F 46224928 Ki = 0.5012 nM T47094 CT3VI4 46224962 Ki = 0.7943 nM T47094 CZ5T6V 46227360 Ki = 3.7 nM T47094 CWC4L2 46227361 Ki = 0.52 nM T47094 CZ61KI 46227362 Ki = 0.1 nM T47094 C37HPA 46227363 Ki = 0.25 nM T47094 CS18JY 46830287 IC50 = 0.1 nM T47094 CI47VS 46881600 IC50 = 0.3 nM T47094 CZ3QW9 46881682 IC50 = 0.04 nM T47094 CUIP97 46881727 IC50 = 0.06 nM T47094 CRD35V 46881728 IC50 = 0.13 nM T47094 CJ7LE6 46881729 IC50 = 2.7 nM T47094 C8LC0K 46881779 IC50 = 0.06 nM T47094 C9ZU7C 46881820 IC50 = 0.07 nM T47094 CIU34R 46881821 IC50 = 1.83 nM T47094 CH7N3A 46883823 IC50 = 0.16 nM T47094 CQPH73 46883824 IC50 = 0.18 nM T47094 C2ZNH5 46883879 IC50 = 0.041 nM T47094 C20UHZ 46884430 IC50 = 0.013 nM T47094 COD4M3 46884431 IC50 = 0.93 nM T47094 CA0JR5 46884432 IC50 = 1.8 nM T47094 C7RKV0 46884433 IC50 = 2 nM T47094 CVKD91 46884434 IC50 = 0.39 nM T47094 CXC50K 46884467 IC50 = 0.11 nM T47094 CI8A2H 46884468 IC50 = 0.51 nM T47094 CN8GC4 46884469 IC50 = 1.1 nM T47094 CY15SL 46884470 IC50 = 0.27 nM T47094 CF1G6L 46884471 IC50 = 0.18 nM T47094 C7KW3I 46884472 IC50 = 2.3 nM T47094 CD46ME 46884473 IC50 = 0.16 nM T47094 CL2E8W 46884515 IC50 = 0.15 nM T47094 C9DMJ2 46884516 IC50 = 0.13 nM T47094 C8BY7G 46884517 IC50 = 1.9 nM T47094 CR04GS 46884518 IC50 = 0.11 nM T47094 CVJ9M0 46884519 IC50 = 5.6 nM T47094 C63IRV 46889466 Ki = 3.05 nM T47094 CZS8I3 46889667 Ki = 1.38 nM T47094 C91JMT 46889668 Ki = 1.72 nM T47094 C7I4CK 46889669 Ki = 2.62 nM T47094 C9FM0R 46889690 Ki = 0.86 nM T47094 C0FBN7 46889691 Ki = 11.1 nM T47094 CLT23D 46889692 Ki = 2.27 nM T47094 C3VA6U 46889693 Ki = 1 nM T47094 C8ZO3Y 46889694 Ki = 1.58 nM T47094 CO39TW 46889695 Ki = 0.51 nM T47094 CPSE79 46889696 Ki = 0.61 nM T47094 CPYO39 46889697 Ki = 0.91 nM T47094 CO1R8E 46889698 Ki = 1.58 nM T47094 CZ0G6A 46947062 IC50 = 0.061 nM T47094 CTQB24 49799942 IC50 = 130 nM T47094 C9M7FZ 49863731 Ki = 0.0053 nM T47094 C9PCU7 49863732 Ki = 0.18 nM T47094 C92LUS 49863733 Ki = 59 nM T47094 C97UJR 49863734 Ki = 1.9 nM T47094 C6HV0T 51002938 Ki = 0.08128 nM T47094 COI28R 51002992 Ki = 0.2754 nM T47094 C2QM9R 51002993 Ki = 0.1175 nM T47094 C8VH5W 51002995 Ki = 0.3236 nM T47094 C6R0ZK 51002996 Ki = 0.1698 nM T47094 CE3Z6R 51003053 Ki = 0.2089 nM T47094 CJQ94A 51003055 Ki = 0.9333 nM T47094 CL39HG 51003056 Ki = 0.1778 nM T47094 C5EWV3 51003117 Ki = 0.6457 nM T47094 CL1DU3 51003118 Ki = 0.1413 nM T47094 C65OHC 51003119 Ki = 0.1995 nM T47094 CMZH79 51003178 Ki = 0.4365 nM T47094 C93GXR 51003494 Ki = 340 nM T47094 CD2YU8 51351496 Ki = 2200 nM T47094 C2UG4W 51351504 Ki = 1600 nM T47094 CE8J6X 52932923 Ki < 0.1585 nM T47094 CYP7K5 52933155 Ki = 0.1 nM T47094 CW1LN2 52937270 Ki = 387 nM T47094 CBRO49 52937271 Ki = 27 nM T47094 C6YJ4V 52937273 Ki = 32 nM T47094 CU43ES 52937467 Ki = 0.5 nM T47094 CE0P8R 52940877 Ki = 1.13 nM T47094 COMU84 52940879 Ki = 0.6 nM T47094 CO2P1X 52940937 Ki = 0.28 nM T47094 C5ETK3 52941351 IC50 = 0.08 nM T47094 CM0IX9 52941489 IC50 = 3.2 nM T47094 CB6X3L 52941506 IC50 = 1.5 nM T47094 C3B1SG 52941550 IC50 = 0.66 nM T47094 CQ68FR 52941570 IC50 = 13 nM T47094 C4QSG6 52942011 Ki = 0.34 nM T47094 C30HVD 52942012 Ki = 0.4 nM T47094 C42BOI 52942803 IC50 = 0.14 nM T47094 CQX80G 52943089 Ki = 1.4 nM T47094 C9LF4T 52943090 Ki = 2.1 nM T47094 CEWV29 52943331 Ki = 0.26 nM T47094 C4OW6U 52943348 Ki = 0.56 nM T47094 CL21TD 52943450 Ki = 0.35 nM T47094 CI71TX 52943848 IC50 = 0.066 nM T47094 CM36DN 52943994 IC50 = 0.11 nM T47094 C7RCO3 52945787 Ki = 0.33 nM T47094 C8UN7I 52946726 Ki = 1.1 nM T47094 C8ME4S 52946917 Ki = 0.37 nM T47094 CW3DA7 52946919 Ki = 0.9 nM T47094 CLZ0T6 52947014 Ki = 0.26 nM T47094 CH7X9N 52947645 IC50 = 1 nM T47094 CSTN95 52947646 IC50 = 0.14 nM T47094 CA3UB6 52947647 IC50 = 0.17 nM T47094 C6LSO0 52948590 IC50 = 0.09 nM T47094 CZ03EM 52948868 IC50 = 0.21 nM T47094 C74IUF 52948931 IC50 = 0.16 nM T47094 C59MTN 52949509 Ki = 1.03 nM T47094 C3VMQ5 52949827 IC50 = 0.77 nM T47094 CLP91C 53249015 IC50 = 4.8 nM T47094 CHB6G2 53320128 Ki = 0.1995 nM T47094 C1VF4P 53379507 IC50 = 6.6 nM T47094 CXL03D 53379508 IC50 = 0.34 nM T47094 CP85ZU 53379509 IC50 = 0.42 nM T47094 CK1C9O 53472113 Ki = 1258.93 nM T47094 C17TLV 54580277 IC50 = 41 nM T47094 C9WA4S 54581251 IC50 = 270 nM T47094 C41TGL 54581252 IC50 = 91 nM T47094 CUH4E9 54581461 Ki = 0.95 nM T47094 CW4Q1K 54582277 IC50 = 653 nM T47094 CJO80U 54582278 IC50 = 235 nM T47094 C6YK5W 54582296 IC50 = 52 nM T47094 CFS4L2 54582297 IC50 = 57 nM T47094 CEFT05 54583959 Ki = 1900 nM T47094 C6OH3G 54584234 IC50 = 279 nM T47094 CN80IV 54585202 IC50 = 53 nM T47094 CGQI45 54585203 IC50 = 434 nM T47094 C0NRK5 54585204 IC50 = 698 nM T47094 CTV97Q 54585205 IC50 = 53 nM T47094 CF6Q9A 54586136 IC50 = 98 nM T47094 C2DYV1 54587142 IC50 = 342 nM T47094 CG2Q8M 54587143 IC50 = 32 nM T47094 CZ56XG 56657842 IC50 = 28 nM T47094 CN2J0U 56658036 IC50 = 9.5 nM T47094 C0AD5O 56661421 IC50 = 77 nM T47094 CT3NM0 56661423 IC50 = 4.9 nM T47094 CT27CV 56662745 IC50 = 1.1 nM T47094 CVP01T 56665366 Ki = 13 nM T47094 CBU60M 56666212 IC50 = 15 nM T47094 C0D1EI 56668295 IC50 = 46 nM T47094 CKT8H2 56668399 IC50 = 3.1 nM T47094 C78VUH 56668401 IC50 = 0.81 nM T47094 CE7K6X 56668794 Ki = 6.8 nM T47094 CXSB71 56671762 IC50 = 97 nM T47094 C9GIX8 56671764 IC50 = 97 nM T47094 CJ0BD7 56671766 IC50 = 280 nM T47094 CC5OX2 56671913 IC50 = 4 nM T47094 C5M3BZ 56675185 IC50 = 220 nM T47094 C8MG3P 56675290 IC50 = 55 nM T47094 C09YQD 56675494 IC50 > 1000 nM T47094 C8Y1QO 56678486 IC50 = 6.1 nM T47094 CCP09Q 56678621 IC50 = 14 nM T47094 C1ON2J 56681830 IC50 = 31 nM T47094 C2X1QE 56681832 IC50 = 270 nM T47094 C8J7IG 56681948 IC50 = 18 nM T47094 COUB01 56681950 IC50 = 2.3 nM T47094 C08AKH 56682292 Ki = 31 nM T47094 CA9F2M 57390403 IC50 = 0.13 nM T47094 C87BKP 57390405 IC50 = 0.054 nM T47094 C7CDR5 57391132 Ki = 158000 nM T47094 C02MLR 57391133 Ki = 100000 nM T47094 CNK2G6 57391771 IC50 = 0.02 nM T47094 C6C1DG 57391807 IC50 = 0.064 nM T47094 C53NEF 57392804 Ki = 0.05012 nM T47094 CZH5A7 57393953 IC50 = 1.9 nM T47094 CO8VD4 57393955 IC50 = 0.1 nM T47094 CH3BG0 57394644 Ki = 79000 nM T47094 CBT8F0 57395686 IC50 = 4.8 nM T47094 CUYS51 57395687 IC50 = 3.7 nM T47094 C90NHR 57395688 IC50 = 0.054 nM T47094 CNDX20 57395691 IC50 = 0.081 nM T47094 C5GOU0 57395693 IC50 = 0.057 nM T47094 C3AX9G 57395695 IC50 = 0.025 nM T47094 C3I2PJ 57396275 Ki = 0.07943 nM T47094 C9AIN2 57396389 Ki = 40000 nM T47094 CT76LK 57397000 IC50 = 0.046 nM T47094 CRJH54 57397019 IC50 = 5.6 nM T47094 C1SBM6 57397020 IC50 = 2.7 nM T47094 COW17K 57397021 IC50 = 0.18 nM T47094 CR79BO 57397022 IC50 = 0.048 nM T47094 CGZ78J 57397481 IC50 = 0.086 nM T47094 C9N6IC 57397483 IC50 = 0.056 nM T47094 CTY0J1 57398076 Ki < 0.1585 nM T47094 C7O9FQ 57398780 IC50 = 2.6 nM T47094 CG5O7I 57398781 IC50 = 3.2 nM T47094 COG59Y 57398782 IC50 = 0.098 nM T47094 C5PF0M 57398783 IC50 = 0.052 nM T47094 CWT5F6 57398784 IC50 = 0.043 nM T47094 CU60RA 57398785 IC50 = 0.11 nM T47094 CQZG19 57399170 IC50 = 1.2 nM T47094 CI0NT2 57399171 IC50 = 0.093 nM T47094 C5RX0C 57400460 IC50 = 2.6 nM T47094 CMT8I0 57400915 IC50 = 0.16 nM T47094 CU9ZB8 57400917 IC50 = 0.049 nM T47094 C43NFV 57400919 IC50 = 0.044 nM T47094 CN0BS4 57400921 IC50 = 0.057 nM T47094 CK2OE6 57400923 IC50 = 0.084 nM T47094 C4VDL3 57402221 IC50 = 0.2 nM T47094 CH5P1G 57402264 IC50 = 0.032 nM T47094 C5HLG6 57402265 IC50 = 0.21 nM T47094 CX09AW 57402266 IC50 = 0.073 nM T47094 C5K3ZP 57402688 IC50 = 0.31 nM T47094 CO1PZ3 57402689 IC50 = 0.17 nM T47094 C1V3UF 57402690 IC50 = 0.075 nM T47094 CF15SP 57402692 IC50 = 0.2 nM T47094 C10WAF 57403249 Ki = 0.0631 nM T47094 C2ONA4 57403990 IC50 = 12 nM T47094 C7JK2N 57403991 IC50 = 0.14 nM T47094 C6ICZ0 57403992 IC50 = 0.035 nM T47094 C3J9UN 57565074 IC50 = 2 nM T47094 C3CDR0 69581370 IC50 = 1.4 nM T47094 CIC7K2 70682893 IC50 = 496 nM T47094 C8Q7NH 70689371 Ki = 56 nM T47094 CLA13H 70693392 IC50 = 95 nM T47094 CLN40O 71449072 IC50 = 0.8 nM T47094 C9DO0T 71449074 IC50 = 35 nM T47094 CCE72K 71449092 Ki = 48000 nM T47094 CU65NS 71449143 IC50 = 2.7 nM T47094 C4D8GV 71450855 IC50 = 220 nM T47094 C21ILJ 71450870 IC50 = 0.3 nM T47094 C6WEU0 71450941 IC50 = 1 nM T47094 C3DW2Y 71450949 IC50 = 164 nM T47094 C7PK5T 71452185 Ki = 0.7 nM T47094 C2MA1K 71452663 IC50 = 16 nM T47094 CBX3C5 71452678 IC50 = 6 nM T47094 CUR6J9 71452815 IC50 = 39 nM T47094 C71KGJ 71453994 Ki = 1.3 nM T47094 CQ82SD 71455736 Ki = 1.4 nM T47094 C8RCG9 71456198 IC50 = 13 nM T47094 C73NUI 71456209 IC50 = 0.08 nM T47094 CQV65R 71456210 IC50 = 133 nM T47094 CC1XL3 71457524 Ki = 1.4 nM T47094 C18VLH 71458000 IC50 = 250 nM T47094 C6H2WN 71458099 IC50 = 86 nM T47094 CL2S4D 71458106 Ki = 0.631 nM T47094 C2C0MK 71458131 IC50 = 3.6 nM T47094 CG7Q5D 71460015 Ki < 3162.28 nM T47094 CUXL38 71461646 Ki = 1.7 nM T47094 CN8CM1 71533722 Ki = 12589.25 nM T47094 CR7E4G 71541370 IC50 = 430 nM T47094 C9IE3U 71541371 IC50 = 480 nM T47094 CFO83N 71541372 IC50 = 74 nM T47094 CI6J5K 71541373 IC50 = 1.9 nM T47094 CC7YB2 71541376 IC50 = 700 nM T47094 CWT0Y3 71541468 IC50 = 12 nM T47094 CGJ86B 71541469 IC50 = 16 nM T47094 C0CBT4 71541470 IC50 = 29 nM T47094 CQ8JN9 71541471 IC50 = 39 nM T47094 CZV7N9 71541472 IC50 = 9.1 nM T47094 CL20CV 71541473 IC50 = 8.7 nM T47094 C6J9NY 71541572 IC50 = 5.3 nM T47094 CS0J6B 71541573 IC50 = 5.3 nM T47094 C5CO8Z 71541574 IC50 = 1.8 nM T47094 CI90PK 71541575 IC50 = 290 nM T47094 C4FS8Z 71541576 IC50 = 11 nM T47094 CSI37G 71541577 IC50 = 6.4 nM T47094 C5D6IE 71541687 IC50 = 3.7 nM T47094 CV47CJ 71549769 Ki = 12589.25 nM T47094 CQ3L2J 71583092 IC50 = 57 nM T47094 CD0P5Z 71583093 IC50 = 1700 nM T47094 CER9H2 71583094 IC50 = 16 nM T47094 CK51UY 71583095 IC50 = 410 nM T47094 CJ8TH9 71583096 IC50 = 110 nM T47094 CC85VD 71583203 IC50 = 660 nM T47094 CI0GU8 71660496 IC50 > 48500 nM T47094 CW0MV2 71716116 Ki = 1 nM T47094 CT82XD 71717930 Ki = 120 nM T47094 CMI1V5 71720664 IC50 = 3.6 nM T47094 CMZ94S 71818133 Ki = 0.066 nM T47094 CAMG13 71818134 Ki = 0.097 nM T47094 CZM8U6 71818277 Ki = 0.0057 nM T47094 C48FZQ 72203985 Ki = 0.138 nM T47094 CL3J7I 72734611 Ki = 2.2 nM T47094 CP5HC1 73212363 Ki > 10000 nM T47094 C86LGQ 73212437 Ki = 15.85 nM T47094 C6DXY3 73212439 Ki = 100 nM T47094 C83GFJ 73212440 Ki = 251.19 nM T47094 CR36KA 73212441 Ki > 10000 nM T47094 C1Y6IU 73212515 Ki = 79.43 nM T47094 CA64UI 73212516 Ki = 316.23 nM T47094 CFC47O 73212517 Ki = 316.23 nM T47094 CG9JP6 73212518 Ki = 251.19 nM T47094 CU30GO 73212519 Ki = 794.33 nM T47094 CE9R0Y 73212588 Ki > 10000 nM T47094 CEU1C3 73212589 Ki > 10000 nM T47094 CKT46G 73212590 Ki > 10000 nM T47094 C7Q1UP 73212591 Ki > 100000 nM T47094 CGU23K 73212592 Ki = 2511.89 nM T47094 C0K4EH 73212593 Ki = 2511.89 nM T47094 C2Q3ZF 73345476 Ki = 2500 nM T47094 CEA84Y 73347011 Ki = 72000 nM T47094 CQ0MH3 73348495 Ki = 0.41 nM T47094 CI69LT 73348949 Ki = 2.6 nM T47094 C8A1DU 73350088 Ki > 100000 nM T47094 CQ0J3N 73350089 Ki = 120 nM T47094 CVR35O 73350234 Ki = 79 nM T47094 C4SKT9 73351579 Ki = 8000 nM T47094 CPS80N 73351736 Ki = 110 nM T47094 C65ZSO 73352606 IC50 = 0.17 nM T47094 C5BPU2 73352970 IC50 = 44 nM T47094 CO25EH 73353047 Ki = 18000 nM T47094 C7PK2H 73353048 Ki > 100000 nM T47094 C9XO0L 73354483 IC50 = 85 nM T47094 CN8D6S 73354569 Ki > 100000 nM T47094 C9FVI0 73354570 Ki = 120 nM T47094 CU9WL2 73354719 Ki = 23 nM T47094 C7O5MI 76311027 IC50 = 93 nM T47094 CZJH91 76314659 IC50 = 470 nM T47094 CB5KG6 76314660 IC50 = 16 nM T47094 CB45FG 76317390 Ki = 12.59 nM T47094 CRMT56 76318226 IC50 = 350 nM T47094 C62AXF 76318227 IC50 = 14 nM T47094 C3B0YJ 76325557 IC50 = 120 nM T47094 CQJ13A 76325558 IC50 = 120 nM T47094 CN52UF 76332768 IC50 = 48 nM T47094 C0B3HG 76332769 IC50 = 38 nM T47094 C9ZMB0 76336391 IC50 = 74 nM T47094 CD5W6K 90417914 Ki = 7943.28 nM T47094 C7E2NA 90644603 Ki = 125.89 nM T47094 CGYH84 90644605 Ki = 199.53 nM T47094 CU3KJ2 90644607 Ki = 50.12 nM T47094 C6OXD3 90644609 Ki = 398.11 nM T47094 C5OXI0 90644611 Ki = 630.96 nM T47094 CI0P4O 90644613 Ki = 125.89 nM T47094 CN3EA2 90644615 Ki = 398.11 nM T47094 CQ84WX 90644617 Ki = 630.96 nM T47094 C5D2IJ 90644619 Ki = 19.95 nM T47094 CW2LI9 90644621 Ki = 63.1 nM T47094 C8O9CH 90644623 Ki = 251.19 nM T47094 C13NEK 90644625 Ki = 316.23 nM T47094 CI46TV 90644627 Ki = 15.85 nM T47094 CGR64B 90644629 Ki = 39.81 nM T47094 CTQD75 90644630 Ki = 19.95 nM T47094 C4UYZ6 90644631 Ki = 31.62 nM T47094 C1GRO9 90644632 Ki = 15.85 nM T47094 C2CRO1 90644633 Ki = 2.512 nM T47094 C58BJM 90644634 Ki = 3.981 nM T47094 C4TYO9 90664465 IC50 = 0.012 nM T47094 CX0B9M 90665209 IC50 = 8.4 nM T47094 C9ZUP4 91809194 IC50 > 10000 nM T47094 CCY0O2 100951644 IC50 = 71000 nM T47094 CNS4V9 102531123 IC50 > 10000 nM T47094 CXL57K 102531124 IC50 > 10000 nM T47094 CY8R0C 102531125 IC50 > 10000 nM T47094 C0OSW4 102531127 IC50 > 10000 nM T47094 C8Z6QX 118722856 IC50 = 16.5 nM T47094 CH5K7Q 118722857 IC50 = 60.6 nM T47094 CRFE13 118722858 IC50 = 9 nM T47094 C2UP4Q 118730932 Ki = 59.7 nM T47094 CGF52A 118730933 Ki = 6.44 nM T47094 CWU0T3 118730934 Ki = 34.7 nM T47094 CT70ZF 118730935 Ki = 3000 nM T47094 CXNT58 118730936 Ki = 1530 nM T47094 CAP2J3 118731113 Ki = 6190 nM T47094 CL6D3T 118731114 Ki = 35 nM T47094 CM35DA 118731115 Ki = 1020 nM T47094 CU9O6M 118731116 Ki = 743 nM T47094 CVT0J9 118731117 Ki = 308 nM T47094 CZ3A0Q 118731118 Ki = 734 nM T47094 CEUG05 118731119 Ki = 16050 nM T47094 CVH6E0 122187205 Ki = 0.34 nM T47094 CP20LG 122187206 Ki = 0.004 nM T47094 C7JS5O 122187722 Ki = 0.47 nM T47094 C27RVE 122187723 Ki = 0.2 nM T47094 CTO0D6 122187724 Ki = 0.016 nM T47094 CJ8D0B 122187725 Ki = 0.85 nM T47094 C76XAE 125111645 IC50 > 10000 nM T47094 CW82BM 127030411 Ki = 1.1 nM T47094 CXK58G 127031644 Ki = 1.4 nM T47094 C1KCW3 127032533 Ki = 0.99 nM T47094 CR4AL9 127032846 Ki = 2.2 nM T47094 C69CGU 127033167 Ki = 1.2 nM T47094 C3L5VD 127033168 Ki = 1.9 nM T47094 CW0D8S 127033173 Ki = 1.4 nM T47094 CO4N2F 127034660 IC50 > 10000 nM T47094 CNQ2Y4 127034696 IC50 > 10000 nM T47094 CRAC83 127034748 IC50 > 10000 nM T47094 CV9Z2G 127034749 IC50 > 10000 nM T47094 CJ7T9U 127034767 IC50 > 10000 nM T47094 CE9Z2Y 127034768 IC50 > 10000 nM T47094 C7CYF5 127034769 IC50 > 10000 nM T47094 CNX2F4 127034928 IC50 > 10000 nM T47094 CATQ52 127034940 IC50 > 10000 nM T47094 CL6OW2 127035038 IC50 > 10000 nM T47094 C1AG9R 127035039 IC50 > 10000 nM T47094 C8WXA7 127035040 IC50 > 10000 nM T47094 CE62OX 127035105 IC50 > 10000 nM T47094 CHAS82 127035106 IC50 > 10000 nM T47094 CJR2D5 127035222 IC50 > 10000 nM T47094 C52ALH 127035367 IC50 > 10000 nM T47094 C2S8IW 127035368 IC50 > 10000 nM T47094 CUV12X 127035512 IC50 > 10000 nM T47094 C9PDL3 127035576 IC50 > 10000 nM T47094 CS78HG 127035706 IC50 > 10000 nM T47094 C2PL6V 127036728 IC50 > 10000 nM T47094 CFC05Q 131954513 Ki = 650 nM T47094 CM1A7G 135405092 IC50 = 0.23 nM T47094 CQJ3E7 135406581 IC50 = 0.07 nM T47094 C59TSQ 135416054 Ki = 0.5 nM T47094 CU05KV 135419433 IC50 = 0.1 nM T47094 CE16KY 135430679 IC50 = 0.42 nM T47094 C1JKC0 135430775 IC50 = 0.43 nM T47094 C1Y3IB 135449286 IC50 = 0.09 nM T47094 CFE46V 135480369 IC50 = 1.7 nM T47094 C6UT1Q 135485796 IC50 = 0.09 nM T47094 C9QR7L 135529973 IC50 = 0.27 nM T47094 CJK8C3 135530616 Ki = 15.85 nM T47094 CAR9K8 135547943 IC50 = 0.09 nM T47094 C2A0TB 135767968 IC50 = 2.2 nM T47094 CYO78E 135890952 IC50 = 19 nM T47094 CM9G7A 136043848 IC50 = 2 nM T47094 CC0D7E 136043849 IC50 = 4.9 nM T47094 CYQM76 136043853 IC50 = 4.7 nM T47094 CA83VQ 136094778 IC50 = 0.61 nM T47094 C7QH2W 136094860 IC50 = 0.56 nM T47094 C6AK3J 136094861 IC50 = 0.1 nM T47094 CE8PS9 136094863 IC50 = 0.1 nM T47094 CE7R1S 136180337 IC50 = 2.4 nM T47094 C3OVA7 136180338 IC50 = 2 nM T47094 CTP08U 136180339 IC50 = 1.5 nM T47094 CL5RJ7 136180340 IC50 = 0.8 nM T47094 CZ82RG 145948744 Ki = 2.2 nM T47094 C3EWL2 145948797 Ki = 1.4 nM T47094 CMD58S 145948809 Ki = 3.3 nM T47094 C2RLY9 145948839 Ki = 2.6 nM T47094 CGA46O 145948847 Ki = 1 nM T47094 CHGW16 145948955 Ki = 3.4 nM T47094 C7N5LP 145948965 Ki = 2.5 nM T47094 CH49XK 145948968 Ki = 5.6 nM T47094 C5E2QA 145948981 Ki = 2.9 nM T47094 CW8QJ9 145964453 IC50 = 200000 nM T47094 C2EC5A 145971823 EC50 = 350000 nM T47094 C72EFN 155551678 Ki = 1.3 nM T47094 CX0EM1 10344874 IC50 = 830 nM T47094 C6RC0T 10552479 Ki = 1560 nM T47094 CLFJ03 10721590 Ki = 77.6 nM T47094 C8GM1T 44337578 IC50 = 100000 nM T47094 C2RQK0 44337620 IC50 = 800 nM T47094 CVL7I1 44337703 IC50 = 2700 nM T47094 CJ63FA 44337704 IC50 = 60600 nM T47094 CI6E1K 44375315 IC50 = 590 nM T47094 CCKO52 44375712 IC50 > 100000 nM T47094 D00HUY 10473960 IC50 = 67 nM T47094 D01NPA 5311311 Ki = 630 nM T47094 D03TPY 9885123 IC50 > 10000 nM T47094 D04TXE 5311350 IC50 = 10000 nM T47094 D05ETM 5311057 IC50 = 0.1698 nM T47094 D05ZUX 44207909 Ki >= 1000 nM T47094 D07NNN 5311312 IC50 = 97.5 nM T47094 D08KSJ 24768351 Ki = 0.046 nM T47094 D09NBN 9915428 IC50 = 3000 nM T47094 D0A1DE 10917690 IC50 = 5200 nM T47094 D0C6RQ 24768356 Ki = 1.4 nM T47094 D0CK8C 24768352 Ki = 100 nM T47094 D0G6GC 25129135 Ki = 3.2 nM T47094 D0J3AO 9914897 IC50 = 2200 nM T47094 D0J8SU 36511 EC50 = 0.05754 nM T47094 D0K9GG 132629 EC50 = 24.4 nM T47094 D0L2CT 24768355 Ki = 0.6 nM T47094 D0N3RM 6450815 Ki = 1 nM T47094 D0P0RB 24768354 Ki = 1.6 nM T47094 D0P1XM 9890435 IC50 = 1 nM T47094 D0PN9R 16655023 Ki = 310 nM T47094 D0Q7HG 24768353 Ki = 14 nM T47094 D0Q7MQ 9796216 IC50 = 0.2 nM T47094 D0S9CI 11989776 IC50 > 1000 nM T47094 D0T2RY 9948320 Ki >= 1000 nM T47094 D0T4JO 9871754 IC50 = 0.24 nM T47094 D0TL4O 10053205 IC50 = 0.8 nM T47094 D0UG6N 10650263 IC50 = 19 nM T47094 D0W3XD 16049828 IC50 > 1000 nM T47094 D0XR4J 85169 Ki = 1.5 nM T47094 D0Z6TG 9852253 Ki = 0.1 nM T91661 D07OAC 132663 IC50 = 4 nM T91661 D08LUT 1973 IC50 = 1.7 nM T91661 D0JI1J 5311109 IC50 = 0.5 nM T91661 CW02OU 14978 IC50 = 470 nM T91661 CHZN50 97186 IC50 = 120 nM T91661 C5Q7PG 97297 Ki = 16.3 nM T91661 C2HZY1 97453 IC50 = 210 nM T91661 CNPD32 128252 IC50 = 310 nM T91661 CUF38C 129111 Ki = 300 nM T91661 CFHV62 385306 IC50 = 85000 nM T91661 C0MC1G 393218 IC50 = 150000 nM T91661 CP7L0Q 446940 IC50 = 40 nM T91661 C3Z2WF 467445 IC50 = 100000 nM T91661 CR92LN 940389 Ki = 5040 nM T91661 C65GXN 2188297 Ki = 184 nM T91661 C4RK8O 3010388 IC50 = 24 nM T91661 C48HYD 3056066 IC50 > 10000 nM T91661 CM48OH 3056069 IC50 = 3600 nM T91661 C3MVQ4 3582931 Ki = 19500 nM T91661 C0MYW9 5106754 Ki = 5440 nM T91661 C9G5QW 6560357 IC50 = 1000 nM T91661 CQZ1J8 9798527 IC50 > 100000 nM T91661 C3O2QU 9802216 IC50 = 1.5 nM T91661 C9L3MV 9804143 IC50 = 1 nM T91661 C9XTO6 9806860 IC50 = 25 nM T91661 CZR3N8 9816781 IC50 = 6330 nM T91661 CG5L7Z 9842886 IC50 > 100000 nM T91661 CZF89B 9872551 IC50 = 8.1 nM T91661 CJ02NM 9880031 IC50 = 47 nM T91661 C7K0YO 9886793 IC50 = 68 nM T91661 CMR58E 9900478 IC50 = 11 nM T91661 C0RQX8 9903135 IC50 > 1000 nM T91661 C5N3DF 9910182 IC50 = 3 nM T91661 CC6X3Y 9910652 IC50 = 0.3 nM T91661 CCM0S4 9915713 IC50 = 350 nM T91661 CN38YF 9923148 IC50 = 200 nM T91661 C4RYF9 9938726 IC50 = 367 nM T91661 CW0U7N 9946703 IC50 = 500 nM T91661 C6V8XR 9947511 IC50 = 433 nM T91661 C3KRQ5 9952948 IC50 = 0.8 nM T91661 C26QPZ 9966768 IC50 = 9 nM T91661 CF5E7X 9967834 IC50 = 1500 nM T91661 C5POS6 10002103 IC50 = 53 nM T91661 C4K8LS 10003439 IC50 = 10 nM T91661 CE3LT0 10004031 IC50 = 130 nM T91661 CR36XH 10043090 IC50 = 0.2 nM T91661 CYMV48 10084205 IC50 = 13000 nM T91661 C30AUM 10109774 IC50 > 1000 nM T91661 CR7Y0D 10110515 IC50 = 2230 nM T91661 C87QCH 10131805 IC50 = 30 nM T91661 CG4VI0 10136788 IC50 = 0.47 nM T91661 CQ2P1H 10154451 IC50 = 4170 nM T91661 CS61WD 10157625 IC50 = 650 nM T91661 C52HMQ 10157755 IC50 = 700 nM T91661 C2IXN3 10180415 IC50 = 70 nM T91661 CQ0G2C 10200044 IC50 = 183 nM T91661 C34PEY 10222462 IC50 > 1000 nM T91661 CE23KW 10253331 IC50 = 10 nM T91661 COX43M 10253975 IC50 = 23 nM T91661 CBN6L0 10270557 IC50 = 567 nM T91661 CAU58E 10273318 IC50 = 115 nM T91661 C4HSO5 10291751 IC50 = 114 nM T91661 C1M5TY 10293769 IC50 = 180 nM T91661 CEDF53 10319137 IC50 = 6 nM T91661 CV79GS 10319941 IC50 = 167 nM T91661 CC05FS 10340386 IC50 = 0.6 nM T91661 C6U4EO 10342811 IC50 = 7.5 nM T91661 C9SJI3 10391910 IC50 = 1.4 nM T91661 C4LOY9 10454249 IC50 = 0.1 nM T91661 CUXS75 10501537 IC50 = 45 nM T91661 CI2OU6 10502034 IC50 = 1.5 nM T91661 CWO0E8 10502035 IC50 = 30 nM T91661 CU91TK 10502860 IC50 = 6 nM T91661 C6R2XN 10503787 IC50 = 100 nM T91661 C07WGQ 10524206 IC50 = 100 nM T91661 C8SNZ3 10524597 IC50 = 6500 nM T91661 C8S9IK 10525360 IC50 = 1200 nM T91661 CI1VM8 10525523 IC50 = 250 nM T91661 C2YM0U 10526980 IC50 = 26 nM T91661 CBM97L 10527849 IC50 = 10000 nM T91661 CJY7X6 10528763 IC50 = 1 nM T91661 CPM12H 10530194 IC50 = 2000 nM T91661 CXZ2Q8 10548287 IC50 = 100 nM T91661 CJW5Q1 10549940 IC50 = 0.8 nM T91661 C5JT2N 10550320 IC50 = 450 nM T91661 C9QX2Z 10552221 IC50 = 120 nM T91661 C3RTD7 10572215 IC50 = 44 nM T91661 CIO0V7 10573376 IC50 = 1200 nM T91661 C9WOA4 10573944 IC50 = 47 nM T91661 CS60QF 10593390 IC50 = 1250 nM T91661 C5S0QH 10596865 IC50 = 3 nM T91661 CZX3R7 10620521 IC50 = 3.6 nM T91661 CB0JL6 10621189 IC50 = 25 nM T91661 CTK76E 10624615 IC50 = 775 nM T91661 CS62NY 10624670 IC50 = 1000 nM T91661 CI9R3N 10641488 IC50 = 50 nM T91661 CV6P8Q 10644087 IC50 = 60 nM T91661 C38MAE 10645621 IC50 = 6.3 nM T91661 C5XRG0 10647163 IC50 = 1000 nM T91661 CUE1N6 10663881 IC50 = 320 nM T91661 CX08JF 10664090 IC50 = 40 nM T91661 C6F7OB 10688712 IC50 = 500 nM T91661 CV0CO1 10690486 IC50 = 63 nM T91661 C85VYD 10693329 IC50 = 1 nM T91661 CFIC23 10716099 IC50 = 300 nM T91661 C3USX0 10719187 IC50 = 2.7 nM T91661 CF8U6W 10741429 IC50 = 2800 nM T91661 COCF29 10741609 IC50 = 1.2 nM T91661 COD6L3 10757745 IC50 = 70 nM T91661 C3OD8S 10757852 IC50 = 80000 nM T91661 C23TNI 10780262 IC50 = 1350 nM T91661 C4QU6S 10789092 IC50 = 2.3 nM T91661 CQWE97 10789377 IC50 = 1.5 nM T91661 C2QIB5 10790781 IC50 = 1200 nM T91661 CCD96O 10825497 IC50 = 16500 nM T91661 CJ4XO7 10835751 IC50 = 35 nM T91661 CQ50RY 10835981 IC50 = 9 nM T91661 CIO6B3 10837996 IC50 = 200 nM T91661 CC1FS9 10853255 IC50 = 1000 nM T91661 C2GN0D 10873200 IC50 = 2000 nM T91661 CW5QT7 10874046 IC50 = 22 nM T91661 CX0T1B 10883874 IC50 = 2.5 nM T91661 C9HW1R 10895093 IC50 = 32 nM T91661 C07YMN 10915775 IC50 = 400 nM T91661 CI9NB0 10934454 IC50 > 10000 nM T91661 CJML31 10936762 IC50 = 467 nM T91661 C1Y0QU 10947859 IC50 = 333 nM T91661 CZFR91 10949191 IC50 = 16 nM T91661 C31THN 10959648 IC50 = 40 nM T91661 CW13JL 11015254 IC50 = 36 nM T91661 CT95ME 11023238 IC50 = 1000 nM T91661 CK45QP 11032790 IC50 = 10000 nM T91661 CCPG09 11068015 IC50 = 467 nM T91661 C3NXE9 11075486 IC50 > 10000 nM T91661 CO85JQ 11078474 IC50 = 170 nM T91661 CVJK64 11080258 IC50 = 42 nM T91661 C4S6OI 11080534 IC50 = 15 nM T91661 C8CW2U 11086280 IC50 > 10000 nM T91661 C18OHZ 11140029 IC50 = 773 nM T91661 CTFP10 11142059 IC50 = 10000 nM T91661 CVKA72 11144253 IC50 = 2.8 nM T91661 CWUN25 11152016 Ki > 50000 nM T91661 CLG5S9 11154768 IC50 = 90 nM T91661 CS94ZT 11166690 IC50 = 200 nM T91661 CZ1UM3 11166830 IC50 = 225 nM T91661 C4IAT3 11190539 IC50 = 625 nM T91661 C6IMO0 11224573 IC50 = 288 nM T91661 CEXB78 11234357 IC50 = 49 nM T91661 CF8A6E 11246252 IC50 = 1000 nM T91661 CUG86D 11248173 IC50 = 7100 nM T91661 C0CW8H 11249663 IC50 = 130 nM T91661 C6XZR3 11249902 IC50 = 197 nM T91661 C4LYU8 11257947 IC50 = 60 nM T91661 CBX0T3 11261214 IC50 = 155 nM T91661 C7ZWP0 11270033 IC50 = 250 nM T91661 C1ZR4B 11284297 IC50 = 450 nM T91661 CNK5H1 11293288 IC50 = 51 nM T91661 CWZK09 11304508 IC50 = 8 nM T91661 CANH80 11306409 IC50 = 625 nM T91661 CVXR35 11315470 IC50 = 230 nM T91661 C5E6RU 11317130 IC50 = 19 nM T91661 CX26DA 11326393 IC50 = 3600 nM T91661 CL3K5U 11327309 IC50 = 6900 nM T91661 C0V6QF 11328858 IC50 = 4500 nM T91661 CV1D7R 11329418 IC50 = 1000 nM T91661 CJW10P 11338636 IC50 = 480 nM T91661 CWUZ32 11362564 IC50 = 2900 nM T91661 CBH49X 11375498 IC50 > 1000 nM T91661 CD4NC9 11383079 IC50 = 500 nM T91661 CS0V9K 11383811 IC50 = 1000 nM T91661 C8MU3B 11441411 IC50 = 150 nM T91661 CX06YD 11466251 IC50 > 1000 nM T91661 CTU6S5 11488638 IC50 = 2000 nM T91661 CW81PN 11503432 IC50 = 2 nM T91661 CZKP62 11525639 IC50 = 145 nM T91661 CU6ND2 11553957 IC50 = 4 nM T91661 C6ZUV4 11560926 IC50 = 7 nM T91661 C3G6EI 11568946 IC50 = 5 nM T91661 C0X7CS 11576266 IC50 = 5.3 nM T91661 CCRF72 11576645 IC50 = 210 nM T91661 C02WNF 11581846 IC50 = 600 nM T91661 CCHG75 11583151 IC50 = 4 nM T91661 C0D4RC 11584077 IC50 = 0.2 nM T91661 CM74TJ 11589023 IC50 = 1700 nM T91661 C5ZG3Q 11589934 IC50 = 25 nM T91661 CZW04G 11591027 IC50 = 0.9 nM T91661 C43NUK 11597018 IC50 = 6 nM T91661 C9OU6E 11603956 IC50 = 40 nM T91661 C9B0QK 11612083 IC50 = 7 nM T91661 C08BQT 11618886 IC50 = 3 nM T91661 C07DBI 11619478 IC50 = 2 nM T91661 CMN80K 11625418 IC50 = 0.8 nM T91661 C31ORL 11632895 IC50 = 20 nM T91661 CL8ZE5 11640594 IC50 = 2 nM T91661 C9S0VG 11640733 IC50 = 10 nM T91661 C3X6BR 11640757 IC50 = 16 nM T91661 C9T3RP 11641141 IC50 = 0.5 nM T91661 C70MTA 11648168 IC50 = 300 nM T91661 CWV9H6 11648278 IC50 = 1 nM T91661 C1BV2D 11659530 IC50 > 10000 nM T91661 CSO0E4 11662079 IC50 = 1.3 nM T91661 C42VUS 11662180 IC50 = 38 nM T91661 C8QXG7 11668212 IC50 = 4 nM T91661 C8XOW2 11668838 IC50 = 4000 nM T91661 C9AV6B 11676143 IC50 = 10 nM T91661 CAE82K 11676479 IC50 = 6 nM T91661 C7TL4I 11683339 IC50 = 5 nM T91661 C2COQ9 11683607 IC50 = 3 nM T91661 CQOE62 11689081 IC50 = 6 nM T91661 CL9TD4 11690975 IC50 = 60 nM T91661 CNC4X3 11729078 IC50 = 30 nM T91661 CGL12P 11752435 IC50 > 1000 nM T91661 CM9EY3 11759755 IC50 = 10000 nM T91661 CN25UR 11773064 IC50 = 300 nM T91661 CETG21 11796739 IC50 = 14 nM T91661 C4FK3O 11798407 IC50 = 800 nM T91661 CJD75T 11987868 IC50 = 2 nM T91661 C4M2AK 12675168 Ki = 15100 nM T91661 C3UI8G 21634257 IC50 > 10000 nM T91661 CT6BD8 23646786 IC50 = 20 nM T91661 CU19GW 23646787 IC50 > 1000 nM T91661 C7M3VB 23646788 IC50 = 9 nM T91661 CAE4V5 23646789 IC50 = 120 nM T91661 C0AP1Q 44129656 IC50 = 1300 nM T91661 CFNW98 44194402 IC50 > 20000 nM T91661 CYFK36 44194404 IC50 > 10000 nM T91661 CJ7W4P 44194405 IC50 > 20000 nM T91661 CCRT57 44194497 IC50 > 10000 nM T91661 CL83NT 44194498 IC50 > 10000 nM T91661 CB9YO4 44194499 IC50 > 10000 nM T91661 CY1S6B 44194500 IC50 > 10000 nM T91661 C9AO3R 44194501 IC50 > 20000 nM T91661 C58RGW 44194502 IC50 > 10000 nM T91661 C9CJ4X 44194503 IC50 = 1100 nM T91661 CUT73N 44194591 IC50 > 10000 nM T91661 CKI1Q0 44194592 IC50 > 10000 nM T91661 CJ32BO 44194593 IC50 > 10000 nM T91661 CV85JG 44194594 IC50 > 20000 nM T91661 C4IH8K 44194595 IC50 > 10000 nM T91661 C29HBA 44194596 IC50 > 10000 nM T91661 COZB06 44194597 IC50 > 10000 nM T91661 CP9RB3 44305396 IC50 = 3.4 nM T91661 C0BNI5 44305399 IC50 = 37.7 nM T91661 C3WEQ4 44305445 IC50 = 71 nM T91661 CRSU16 44305631 IC50 = 4.1 nM T91661 CK2UY0 44305632 IC50 = 42.5 nM T91661 C0BX9P 44305633 IC50 = 1.8 nM T91661 CU1XY3 44329981 IC50 = 460 nM T91661 CQI74C 44330022 IC50 = 550 nM T91661 CGH34R 44333528 IC50 = 81.9 nM T91661 CQ3GT2 44333559 IC50 = 22.8 nM T91661 C1XER9 44333577 IC50 = 153.8 nM T91661 CY6ZS8 44333687 IC50 = 7.5 nM T91661 CYO16S 44333688 IC50 = 6.5 nM T91661 CBA8Q1 44333820 IC50 = 43.7 nM T91661 CM46IT 44333863 IC50 = 7.5 nM T91661 CJ1GM4 44334064 IC50 = 10.4 nM T91661 CAK27Q 44334080 IC50 = 2.8 nM T91661 CQ8OT4 44334083 IC50 = 8.3 nM T91661 C4GZ3T 44334090 IC50 = 18.8 nM T91661 CXF0O9 44334106 IC50 = 7.2 nM T91661 C1Y7OR 44334205 IC50 = 7.1 nM T91661 CB6V0N 44362407 IC50 = 1.5 nM T91661 CVZN78 44362550 IC50 = 280 nM T91661 C64TIG 44365982 IC50 = 22000 nM T91661 CK5S2T 44366104 IC50 = 163 nM T91661 CBS4Y7 44386439 IC50 = 60 nM T91661 C9EWB6 44386502 IC50 = 240 nM T91661 C7PSX6 44386547 IC50 = 260 nM T91661 C5AIL9 44386650 IC50 > 10 nM T91661 C9M1BI 44386651 IC50 > 10 nM T91661 C9MLZ0 44386668 IC50 = 200 nM T91661 CC62ZV 44386698 IC50 = 40 nM T91661 C75APM 44386701 IC50 = 90 nM T91661 CH42NY 44386707 IC50 = 1 nM T91661 CAW4I7 44386715 IC50 = 130 nM T91661 CR7S0H 44386750 IC50 > 1 nM T91661 C13DFH 44386751 IC50 = 200 nM T91661 C0YHQ4 44386752 IC50 = 270 nM T91661 CS3LE7 44386754 IC50 = 230 nM T91661 CDJ71I 44386774 IC50 = 70 nM T91661 C2VH7P 44386810 IC50 = 1.5 nM T91661 CFR4T7 44386831 IC50 > 10 nM T91661 C1YHX7 44386848 IC50 = 40 nM T91661 C7KC4U 44386849 IC50 > 1 nM T91661 C64PQD 44386855 IC50 > 10 nM T91661 C4ZA9D 44386859 IC50 > 10 nM T91661 C87HEB 44386910 IC50 = 210 nM T91661 CYHB58 44386912 IC50 = 70 nM T91661 CH9XF1 44386913 IC50 > 10 nM T91661 CGD3O2 44386956 IC50 = 90 nM T91661 C0A2JH 44386973 IC50 > 10 nM T91661 C26CQS 44387016 IC50 > 10 nM T91661 CK16QW 44387024 IC50 = 130 nM T91661 CV91EM 44387025 IC50 = 50 nM T91661 C56ZTO 44387081 IC50 > 10 nM T91661 CRQ3D5 44387125 IC50 = 120 nM T91661 CUY8J1 44387139 IC50 = 30 nM T91661 CMY83G 44387156 IC50 = 70 nM T91661 CNT8H2 44393044 IC50 = 72 nM T91661 C6C7PT 44393070 IC50 = 120 nM T91661 CR29CI 44393087 IC50 = 460 nM T91661 CFA26E 44393112 IC50 = 300 nM T91661 CMT2D4 44393130 IC50 = 22 nM T91661 C3HVR8 44393153 IC50 = 82 nM T91661 C9UMS7 44393160 IC50 > 1000 nM T91661 CC29JG 44393165 IC50 = 100 nM T91661 CEQ3D9 44393166 IC50 = 75 nM T91661 CPU9E2 44393176 IC50 = 82 nM T91661 C4HO6N 44393221 IC50 > 1000 nM T91661 C1QN6V 44399052 IC50 = 20 nM T91661 CKS1P2 44399127 IC50 = 900 nM T91661 C4UZB0 44399203 IC50 = 38 nM T91661 C8ZY7A 44399248 IC50 = 45 nM T91661 C9PF3R 44405185 IC50 = 1.3 nM T91661 CO1M0S 44405195 IC50 = 0.5 nM T91661 CXLK65 44405205 IC50 = 1 nM T91661 CH4K6J 44405222 IC50 = 530 nM T91661 CV01QB 44405223 IC50 = 2500 nM T91661 CP1G9E 44405224 IC50 = 460 nM T91661 C7JZR6 44405231 IC50 = 2500 nM T91661 CX6PQ8 44405232 IC50 = 880 nM T91661 CF0EI7 44405282 IC50 = 27 nM T91661 CRGU57 44405284 IC50 = 380 nM T91661 CBV0Q7 44405285 IC50 = 100 nM T91661 CACI93 44405288 IC50 = 140 nM T91661 CGX35Y 44405297 IC50 = 45 nM T91661 CVFE85 44405300 IC50 = 2 nM T91661 CY63WP 44405302 IC50 = 0.6 nM T91661 CG82KD 44405914 IC50 = 4 nM T91661 CD2TR4 44423484 IC50 = 3 nM T91661 CSM29F 44423485 IC50 = 5 nM T91661 C4DC1A 44423486 IC50 = 300 nM T91661 CG6CS2 44423487 IC50 = 1000 nM T91661 C3Q4KW 44423488 IC50 = 600 nM T91661 C7VK2M 44423489 IC50 > 1000 nM T91661 CS48DL 44423490 IC50 > 1000 nM T91661 CXK6F8 44423491 IC50 > 1000 nM T91661 C80WIN 44423492 IC50 = 100 nM T91661 C94JXQ 44423493 IC50 = 14 nM T91661 CGKR45 44423494 IC50 = 300 nM T91661 CWN8X9 44423495 IC50 > 1000 nM T91661 CFMC50 44423496 IC50 = 80 nM T91661 C9WXM4 44423497 IC50 = 38 nM T91661 CMX79L 44423498 IC50 = 6 nM T91661 CQB65U 44423499 IC50 = 8 nM T91661 C1NDF8 44423500 IC50 = 13 nM T91661 CHJ45S 44423501 IC50 = 75 nM T91661 CS7EW1 44423502 IC50 = 10 nM T91661 C1EFT2 44423503 IC50 = 3 nM T91661 CXD64W 44423504 IC50 = 330 nM T91661 CRD47W 44423505 IC50 = 18 nM T91661 CL9QJ3 44423506 IC50 = 20 nM T91661 C6BI5K 44423507 IC50 = 22 nM T91661 C8SX6M 44423508 IC50 = 16 nM T91661 CT2JL3 44423509 IC50 = 90 nM T91661 C58TAG 44423510 IC50 = 60 nM T91661 CS2QR0 44423511 IC50 = 25 nM T91661 CEP26G 44423512 IC50 = 50 nM T91661 C7P0EA 44423513 IC50 = 216 nM T91661 CG83BU 44423514 IC50 = 500 nM T91661 C4BKM0 44423515 IC50 = 43 nM T91661 C9Y1ZK 44423516 IC50 = 43 nM T91661 CA0GM9 44423517 IC50 = 10 nM T91661 CTN73D 44423518 IC50 = 17 nM T91661 CM5FI4 44423519 IC50 = 8 nM T91661 C78LXW 44423520 IC50 = 700 nM T91661 C4D5MS 44423521 IC50 = 110 nM T91661 CW39GI 44423522 IC50 = 14 nM T91661 C3LT6I 44423523 IC50 = 83 nM T91661 CBED70 44423524 IC50 = 58 nM T91661 CKHY59 44423525 IC50 = 1 nM T91661 C8X5QT 44423526 IC50 = 6 nM T91661 C03FJR 44423527 IC50 = 62 nM T91661 C6QHU5 44423528 IC50 = 39 nM T91661 C53SFE 44423529 IC50 = 9 nM T91661 C5SRZ0 44423530 IC50 = 120 nM T91661 C63ANF 44423531 IC50 = 167 nM T91661 C6MER9 44423532 IC50 = 38 nM T91661 CCG4Q0 44423533 IC50 = 0.4 nM T91661 CA47CD 44423534 IC50 = 1 nM T91661 C6N4AP 44423535 IC50 = 161 nM T91661 C20MTO 44423536 IC50 = 72 nM T91661 CRP80X 44423537 IC50 = 88 nM T91661 CUR41P 44423538 IC50 = 101 nM T91661 CN5GL0 44591776 IC50 > 100000 nM T91661 C2GM0C 44626657 IC50 > 20000 nM T91661 CZTQ89 44626658 IC50 > 10000 nM T91661 C2IQ9C 44626659 IC50 > 10000 nM T91661 C51OKP 44626660 IC50 > 10000 nM T91661 C3P0FK 44626661 IC50 > 10000 nM T91661 C85CEW 44626757 IC50 > 5000 nM T91661 CLUT25 44626758 IC50 > 10000 nM T91661 C78DBH 44626759 IC50 > 10000 nM T91661 CSEL62 44626760 IC50 > 20000 nM T91661 CG83QE 44626761 IC50 > 10000 nM T91661 C1I8TS 44626762 IC50 = 1300 nM T91661 CMT6R0 44626763 IC50 > 20000 nM T91661 C7C4MN 44626851 IC50 = 290 nM T91661 C9KS5F 44626852 IC50 = 1200 nM T91661 CN5XE0 44626853 IC50 = 3400 nM T91661 CP5Q1F 44776615 Ki = 5100 nM T91661 CJ1I8Y 46875861 IC50 = 154881661.9 nM T91661 C6UOZ3 46875866 IC50 = 1000000000 nM T91661 C09CDZ 46875885 IC50 = 741310241.3 nM T91661 CYBT26 46875916 IC50 = 60255958.61 nM T91661 C9SA6G 46876002 Ki = 40 nM T91661 C8E5IO 46876059 Ki = 300 nM T91661 CBG6E4 46876062 Ki = 170 nM T91661 CZIF64 46876066 Ki = 150 nM T91661 CPI93Y 46876067 Ki = 8500 nM T91661 C87DKA 46876070 Ki = 160 nM T91661 CAWV48 49783975 IC50 > 5000 nM T91661 C9HYF4 49783976 IC50 > 5000 nM T91661 CA6Q0G 49784053 IC50 > 10000 nM T91661 CBU14H 49784054 IC50 > 10000 nM T91661 C5BSU4 49784055 IC50 > 5000 nM T91661 CUD3Q6 49784056 IC50 > 2000 nM T91661 CH4EQ1 49784057 IC50 > 5000 nM T91661 CC4R3E 49784058 IC50 > 5000 nM T91661 CEF1T8 49784059 IC50 > 5000 nM T91661 C0NUL6 49784131 IC50 > 10000 nM T91661 C21DQR 49784132 IC50 > 20000 nM T91661 CY6P9N 49784133 IC50 = 4500 nM T91661 C95YUM 49784134 IC50 > 10000 nM T91661 C9K1QF 49784135 IC50 = 200 nM T91661 C2G4IH 49784136 IC50 > 20000 nM T91661 CWZJ21 49784137 IC50 = 2300 nM T91661 CI4UX1 49784203 IC50 > 5000 nM T91661 CL6I8D 49784438 IC50 = 50 nM T91661 C6A1IB 49840765 IC50 > 10000 nM T91661 CQPE91 51349441 IC50 = 3500 nM T91661 CBW43N 51349442 IC50 = 2500 nM T91661 C8KP1E 51349443 IC50 = 12500 nM T91661 CD8HM7 51349444 IC50 = 3200 nM T91661 C53UAO 51349445 IC50 = 1000 nM T91661 C51FEC 51349446 IC50 = 2000 nM T91661 C6G5XP 51349586 IC50 = 4000 nM T91661 CZ13YW 51349587 IC50 = 2500 nM T91661 C3I4LP 51349588 IC50 = 6200 nM T91661 CVY9J2 51349589 IC50 = 6700 nM T91661 CF92ZM 51349590 IC50 = 14000 nM T91661 CCTI31 51349731 IC50 = 15000 nM T91661 C48DXB 51349732 IC50 = 3000 nM T91661 C12FQV 51349733 IC50 = 7500 nM T91661 CT2PF1 51349734 IC50 = 3000 nM T91661 C8NF6U 51349735 IC50 = 14000 nM T91661 C18EGO 51349736 IC50 = 22500 nM T91661 CTX1O7 51349862 IC50 = 10000 nM T91661 CNXO64 51349863 IC50 = 10000 nM T91661 CWK3N0 51349864 IC50 = 10000 nM T91661 C6VD2H 51349865 IC50 = 2500 nM T91661 CK53FN 51349866 IC50 = 11000 nM T91661 CYNG08 51350275 IC50 = 8000 nM T91661 C70VWB 51350276 IC50 = 4500 nM T91661 CLZR64 51350277 IC50 = 3500 nM T91661 COI78N 51350278 IC50 = 7000 nM T91661 CKMC05 51350279 IC50 = 7000 nM T91661 C1H5ZF 51350280 IC50 = 1200 nM T91661 C8IK2L 51350408 IC50 = 2000 nM T91661 CMC75F 51350409 IC50 = 8000 nM T91661 C2YJD0 51350410 IC50 = 200000 nM T91661 CSC9B3 51350411 IC50 = 150000 nM T91661 CO62XQ 51350412 IC50 = 4000 nM T91661 CTSM04 51350413 IC50 = 4400 nM T91661 CEU91N 51350551 IC50 = 5000 nM T91661 CAU15E 51350552 IC50 = 2200 nM T91661 C2OP6D 51350553 IC50 = 2000 nM T91661 C5VSG2 51350674 IC50 = 9000 nM T91661 CZK82O 51351417 IC50 = 1200 nM T91661 C1PLR5 51351418 IC50 = 4500 nM T91661 CYTN06 51351419 IC50 = 1000 nM T91661 C3TCP9 51351420 IC50 = 21400 nM T91661 CP4U6L 53317344 IC50 > 1000000 nM T91661 CES05N 53323895 IC50 = 5260 nM T91661 CFG8P9 53326545 IC50 = 35000 nM T91661 CDA7P5 56671903 IC50 = 13000 nM T91661 CB6WA9 76311328 IC50 = 4400 nM T91661 CE75JG 76314919 IC50 = 5150 nM T91661 C4W9QP 76314920 IC50 = 6350 nM T91661 CG79WR 76314921 IC50 = 300 nM T91661 C7MY4E 76318534 IC50 = 15400 nM T91661 CTAM57 76318535 IC50 > 20000 nM T91661 COJ05B 76318536 IC50 = 2400 nM T91661 CB71YN 76318537 IC50 = 2900 nM T91661 C45YRI 76318538 IC50 = 2100 nM T91661 CYA9S3 76322193 IC50 = 1970 nM T91661 CRCY59 76336669 IC50 = 8350 nM T91661 CBI46H 76336670 IC50 = 3070 nM T91661 CX2B1G 101884764 IC50 > 20000 nM T91661 CQ4C5J 101884765 IC50 > 10000 nM T91661 CON9D7 101884767 IC50 > 20000 nM T91661 CMS25I 101884768 IC50 > 10000 nM T91661 CE79ZX 101884769 IC50 > 20000 nM T91661 CQ0GR4 101884770 IC50 > 10000 nM T91661 CS4GT6 101884771 IC50 > 10000 nM T91661 CTMQ47 101884772 IC50 > 10000 nM T91661 CY0HX7 101884773 IC50 > 20000 nM T91661 C7K3UZ 101884774 IC50 > 20000 nM T91661 C20FIR 118716611 IC50 > 20000 nM T91661 C8XI2A 118716612 IC50 = 3300 nM T91661 C4L7AQ 118716613 IC50 > 20000 nM T91661 C7IZY8 118716614 IC50 > 10000 nM T91661 CBIZ81 118716615 IC50 > 10000 nM T91661 CG8QN5 118716616 IC50 > 10000 nM T91661 CYF82N 134229886 IC50 > 10000 nM T91661 CN9QI1 134229890 IC50 > 10000 nM T91661 CIGR54 134229893 IC50 > 10000 nM T91661 C7SAP0 134229894 IC50 > 10000 nM T91661 CI2RJ6 134229895 IC50 > 10000 nM T91661 C5FTY0 134229898 IC50 = 3940 nM T91661 C05CIH 134229902 IC50 > 10000 nM T91661 C0UQ4T 134229903 IC50 > 10000 nM T91661 CW15HL 134229904 IC50 = 336 nM T91661 CVT10Q 134229909 IC50 > 10000 nM T91661 CK1T6P 134229912 IC50 > 10000 nM T91661 C7FEH6 134229913 IC50 = 300 nM T91661 C8W7FH 134229914 IC50 > 10000 nM T91661 CBEH85 134229916 IC50 > 10000 nM T91661 C1MK8V 134229926 IC50 > 10000 nM T91661 CH1E8V 134229934 IC50 = 7120 nM T91661 CFY73D 134229959 IC50 > 10000 nM T91661 C6HTA7 138105921 Ki > 50000 nM T91661 CNZ7J0 139582257 Ki = 11100 nM T91661 C3VQN6 145964437 IC50 > 50000 nM T91661 CB32OW 145964815 IC50 > 50000 nM T91661 C6HD7A 145966030 IC50 = 31600 nM T91661 C3ITW7 145966076 IC50 = 13700 nM T91661 C4OEW5 145966583 IC50 > 50000 nM T91661 C82GAM 145972125 IC50 = 13600 nM T91661 CV0L6A 145972558 IC50 = 50000 nM T91661 C35LOD 145973081 IC50 > 50000 nM T91661 CZE89S 145974229 IC50 > 50000 nM T91661 CGB7L4 145974437 IC50 = 40000 nM T91661 C43GFI 145975558 IC50 = 13600 nM T91661 CTFJ90 145975836 IC50 > 50000 nM T91661 C40HMI 145976797 IC50 = 57400 nM T91661 CMZ81R 145976977 IC50 = 32200 nM T91661 CD5KI4 145977612 IC50 = 24700 nM T91661 CQ7DM1 145977815 IC50 > 50000 nM T91661 CH02MF 155510479 IC50 = 115 nM T91661 C8SWN4 155514253 IC50 = 114 nM T91661 CR1J0M 155515702 Ki = 410 nM T91661 C6DH5O 155519526 Ki > 50000 nM T91661 C1DYH7 155520128 Ki = 5640 nM T91661 CF3AS8 155520320 Ki > 50000 nM T91661 CYB89F 155524154 IC50 > 10000 nM T91661 C89UZV 155526021 Ki = 9180 nM T91661 CD8M6G 155526553 Ki > 50000 nM T91661 C34SNI 155527835 Ki = 8560 nM T91661 CG09PC 155527924 IC50 = 0.06 nM T91661 CL4Q7C 155529159 IC50 > 10000 nM T91661 CJ4Y7C 155529316 IC50 > 10000 nM T91661 C2BTO7 155530232 Ki = 1600 nM T91661 CA2Z6J 155536078 IC50 = 3340 nM T91661 C6YJ9Q 155537423 Ki > 50000 nM T91661 CUH95R 155537886 Ki > 50000 nM T91661 C8QO7E 155538272 IC50 > 10000 nM T91661 CF09QI 155540931 IC50 > 10000 nM T91661 C7MJ9Y 155541950 IC50 = 6010 nM T91661 C64UFG 155542277 Ki = 25400 nM T91661 CWEP21 155543135 IC50 = 5380 nM T91661 CM67JL 155543219 Ki > 50000 nM T91661 CA4WY5 155543567 Ki > 50000 nM T91661 C3U8IS 155549597 Ki >= 15100 nM T91661 C48ZXQ 155550681 IC50 > 10000 nM T91661 CCN79V 155551943 IC50 > 10000 nM T91661 C9JD0P 155551973 IC50 = 3580 nM T91661 C70JRG 155555792 IC50 = 470 nM T91661 C3DF2T 155556596 IC50 = 140 nM T91661 CP1MH2 155562414 IC50 = 2240 nM T91661 C5VE3W 155562953 IC50 = 110 nM T91661 CQ8GI3 155564053 Ki = 25200 nM T91661 C5TS7Q 155564824 IC50 = 88 nM T91661 C3YF6X 155568904 Ki = 8750 nM T91661 D03SHX 9842606 IC50 = 9 nM T91661 D08AWL 384831 IC50 = 130000 nM T91661 D0H6WV 6245 IC50 = 10000 nM T59679 D00XWD 135409453 EC50 = 1 nM T59679 D04QSJ 3052762 Ki = 2.512 nM T59679 D08VYV 4168 EC50 = 794.33 nM T59679 D0K0KH 656665 Ki = 199.53 nM T59679 D01ABX 71451950 EC50 = 0.8 nM T59679 D01HVZ 11961293 Ki = 0.3981 nM T59679 D02YKI 53354764 Ki = 0.15 nM T59679 D04AHY 1471834 Ki = 72 nM T59679 D04GMY 11842633 EC50 = 0.631 nM T59679 D0X2XF 177336 Ki = 0.05248 nM T59679 D06DZI 107780 Ki < 10000 nM T59679 D08AWI 11430856 Ki > 5000 nM T59679 D0K1SZ 3019427 EC50 = 290 nM T59679 D0U7VZ 11225102 EC50 = 2.512 nM T59679 D0YP7L 6604889 Ki = 1258.93 nM T59679 D0ZG9N 132337 EC50 = 19.95 nM T59679 CZUI83 2769 Ki = 29 nM T59679 C9UO6W 42499 EC50 = 398.11 nM T59679 COE0W7 44575 EC50 = 79.43 nM T59679 CKP25M 121881 Ki = 0.01585 nM T59679 CF1O8E 130946 Ki = 13 nM T59679 C0B2ZX 182592 IC50 = 49 nM T59679 CVZW19 182593 Ki = 31.62 nM T59679 CE13LW 203435 EC50 = 251.19 nM T59679 CW38FP 5311047 EC50 = 19.95 nM T59679 C3A1FO 6604789 Ki = 251.19 nM T59679 C0QCK1 6918455 Ki = 3981.07 nM T59679 CD0Z4I 6918648 Ki = 3162.28 nM T59679 CXI72O 9799010 EC50 = 39.81 nM T59679 C7AFR2 9800656 Ki = 1 nM T59679 C8VC5R 9807895 Ki = 0.05012 nM T59679 CJ90UH 9817713 Ki = 316.23 nM T59679 C3WSY6 9839803 Ki = 63.1 nM T59679 CM13ZV 9856041 Ki = 1800 nM T59679 CAQ9L7 9869791 Ki = 0.2512 nM T59679 C1DWJ6 9870390 Ki = 0.05012 nM T59679 C9BW8Z 9870916 Ki = 0.03162 nM T59679 CY20GO 9873926 Ki = 0.03162 nM T59679 CKLR65 9882676 EC50 = 125.89 nM T59679 CS16EH 9886435 Ki = 0.7943 nM T59679 C3J8GU 9892409 Ki < 7943.28 nM T59679 C5ZDX7 9892465 Ki = 0.0631 nM T59679 C89DSU 9892494 Ki = 0.03162 nM T59679 CUD0A3 9912434 Ki = 0.3981 nM T59679 C78MDV 9913554 Ki = 5011.87 nM T59679 C6UN1R 9914629 Ki = 0.02512 nM T59679 CY3FW6 9924349 Ki = 169 nM T59679 CWO45F 9935387 Ki = 1584.89 nM T59679 C7XA3G 9936969 Ki = 0.01585 nM T59679 CYH3R7 9947817 Ki = 2400 nM T59679 CC82OS 9950216 IC50 < 10 nM T59679 C3ZQN6 9954930 Ki = 0.07943 nM T59679 CSM53Z 9975257 EC50 = 72.44 nM T59679 CK18LT 10020895 Ki = 4000 nM T59679 C6VO4P 10046170 Ki > 1000 nM T59679 C2JZL1 10048222 IC50 > 1000 nM T59679 C3E5CB 10337773 Ki = 398.11 nM T59679 C9IAV3 10346043 Ki = 3162.28 nM T59679 CTZ5U9 10347130 Ki = 64 nM T59679 C69KIB 10385855 IC50 > 10000 nM T59679 C08RCI 10408029 Ki = 12.5 nM T59679 C4TPN1 10413595 Ki = 3981.07 nM T59679 CD7U5I 10433930 Ki > 10000 nM T59679 CIE39G 10493462 EC50 = 199.53 nM T59679 CP8NL9 10521792 EC50 = 14 nM T59679 CM9L0P 10524522 Ki = 1.4 nM T59679 CJ2Q4D 10526438 Ki = 9.8 nM T59679 C4AU3Q 10548505 Ki = 1.4 nM T59679 CCD47O 10550242 Ki = 296 nM T59679 CHE80N 10573876 Ki < 6309.57 nM T59679 CC4PJ9 10623729 Ki = 199.2 nM T59679 C0VY3W 10643698 EC50 = 31.62 nM T59679 C4N0RK 10644148 Ki = 1.5 nM T59679 C90VMP 10645103 Ki = 16.8 nM T59679 CF0ZO5 10645984 Ki = 162 nM T59679 CL8F7P 10666935 Ki = 6.7 nM T59679 C89LQT 10669143 Ki = 23.1 nM T59679 C17GBZ 10669778 Ki = 17.7 nM T59679 C6IPX1 10688893 Ki = 91.9 nM T59679 CP8B5F 10715463 Ki = 3.5 nM T59679 CLHS38 10716689 Ki > 1000 nM T59679 CBK4G2 10717193 Ki = 715 nM T59679 C95UEV 10739944 Ki = 11.5 nM T59679 CL7SM2 10741078 Ki = 2 nM T59679 CCJ98P 10781509 Ki > 1000 nM T59679 CL42IU 10811181 Ki = 240 nM T59679 C4PK2F 10812045 Ki = 64 nM T59679 CY3Q6I 10828801 EC50 = 316.23 nM T59679 CY89HI 10830094 Ki > 1000 nM T59679 CD4G1Z 10834000 Ki = 23 nM T59679 C8MHZ9 10835110 Ki < 3162.28 nM T59679 C6HMZ7 10836823 Ki > 1000 nM T59679 CILH21 10897011 Ki = 264 nM T59679 CC0V6Y 10919426 Ki = 180 nM T59679 CI18PE 10930618 Ki = 96 nM T59679 CN7KR9 11005668 Ki = 7.5 nM T59679 C0CM3L 11039391 Ki = 116 nM T59679 CG5V8W 11039730 Ki = 31 nM T59679 CDU83T 11050452 Ki = 183 nM T59679 CQG52P 11093246 Ki = 32 nM T59679 C8JR1A 11135810 Ki = 59 nM T59679 CV8H3Y 11146446 Ki = 1720 nM T59679 CVJI40 11146533 Ki = 24 nM T59679 C18JXF 11153975 Ki = 0.1 nM T59679 CZN0I7 11166796 EC50 = 0.38 nM T59679 CLKO85 11168006 EC50 = 3.981 nM T59679 C2CB4G 11174673 Ki = 58 nM T59679 C1BHW0 11293856 Ki = 1.259 nM T59679 CJS9C0 11304851 IC50 > 25000 nM T59679 CSW9T2 11317280 Ki = 0.1585 nM T59679 CS0GR3 11350913 EC50 = 0.5 nM T59679 C7M3XJ 11397742 Ki = 0.1995 nM T59679 CLW3Z1 11432106 EC50 = 10 nM T59679 CV46TC 11498641 Ki = 37 nM T59679 CJ57CQ 11504722 EC50 = 0.3981 nM T59679 CLB78A 11513350 Ki = 7 nM T59679 C67XMT 11519716 EC50 = 0.7943 nM T59679 C02HFE 11520559 Ki = 488 nM T59679 CK0DQ8 11520655 Ki = 10 nM T59679 CHZK27 11527897 Ki = 19 nM T59679 C3T7FD 11549456 Ki = 24 nM T59679 C2RB9L 11557207 Ki = 113 nM T59679 CPC31J 11577105 Ki = 13 nM T59679 CRF3A9 11593090 Ki = 13 nM T59679 CGX8F6 11596869 Ki > 6310000 nM T59679 C89OJE 11600413 Ki = 16 nM T59679 C8N3DH 11606227 EC50 = 0.7943 nM T59679 C8OMW6 11622025 Ki = 20 nM T59679 CQ5TN6 11627949 EC50 = 0.7943 nM T59679 CR6MT3 11629240 Ki = 11 nM T59679 C8RF2N 11629247 Ki = 5 nM T59679 CX51VG 11629268 Ki = 3 nM T59679 CR6IP9 11643822 Ki = 50 nM T59679 CV1A3S 11650641 Ki = 21 nM T59679 C26YBX 11677434 EC50 = 2.512 nM T59679 C74MOI 11686414 Ki = 8 nM T59679 CTRW81 11686484 Ki = 11 nM T59679 CV69DN 11686510 Ki = 200 nM T59679 C1X0UW 11693471 Ki = 9 nM T59679 CJ9ZK2 11714709 Ki = 31 nM T59679 C35YHO 11714901 Ki = 9 nM T59679 C5VX4Q 11794824 Ki = 9.2 nM T59679 C6LZ9U 11796362 Ki = 3 nM T59679 C8WCO2 11813759 Ki = 181 nM T59679 C2FNW4 11813852 Ki = 7 nM T59679 CFA38S 11966400 Ki = 77 nM T59679 CF5P0Q 15485936 Ki = 0.1 nM T59679 CG8KR9 16005860 IC50 = 1400 nM T59679 C2L3QU 17754944 Ki = 34 nM T59679 C5WI8C 17755039 Ki = 44 nM T59679 C1RO4E 17755040 Ki = 18 nM T59679 CBN32C 17755140 Ki = 19 nM T59679 CD9R7T 17755141 Ki = 10 nM T59679 CU6V4S 17756314 Ki = 8 nM T59679 CZ2FX8 17756414 Ki = 40 nM T59679 CY1F5Q 17756415 Ki = 25 nM T59679 C8O0IA 17756519 Ki = 23 nM T59679 CH31QA 17984294 Ki = 0.2512 nM T59679 C10LOR 19081860 EC50 = 15.85 nM T59679 CLA1H6 19081862 EC50 = 39.81 nM T59679 CF7AR1 19081885 EC50 = 12.59 nM T59679 C1MW7J 19081962 EC50 = 63.1 nM T59679 CE1SL2 19081984 EC50 = 10 nM T59679 CQ3JL0 19956256 IC50 = 870.96 nM T59679 C1ZL3W 20030109 EC50 = 63.1 nM T59679 CN85CQ 21252889 Ki = 0.3162 nM T59679 CT4ZC0 21252890 Ki = 7.943 nM T59679 CN1XA4 21252891 Ki = 0.3981 nM T59679 C6AFN2 21252894 Ki = 0.1585 nM T59679 CTUY04 21252899 Ki = 0.631 nM T59679 C2P1TL 21252902 Ki = 0.7943 nM T59679 CUL2W0 21268031 Ki = 0.1259 nM T59679 CTN64B 21268033 Ki = 0.1 nM T59679 CYKE06 21268036 Ki = 0.07943 nM T59679 CCIO21 21268037 Ki = 0.1259 nM T59679 C7ZEF0 24856058 IC50 > 10000 nM T59679 C3HK0J 24865725 Ki > 10000 nM T59679 C0O6FX 24865727 Ki = 7943.28 nM T59679 CM1H6K 25016328 IC50 = 134 nM T59679 CQ28EH 25016330 IC50 = 68 nM T59679 CP6K8J 25024727 IC50 > 10000 nM T59679 C40XJV 42618248 Ki = 5 nM T59679 CK2J5X 42618250 EC50 = 9 nM T59679 CS62YH 42618251 Ki = 12 nM T59679 C0KS9W 42618252 Ki = 2 nM T59679 C03GKH 42646835 Ki = 144.54 nM T59679 C35SCP 44224237 EC50 = 0.3981 nM T59679 CK7F2E 44240743 Ki = 6000 nM T59679 CJX2V5 44247808 EC50 = 39.81 nM T59679 C6ZC7G 44247811 EC50 = 15.85 nM T59679 C9NE7C 44247813 EC50 = 15.85 nM T59679 C0H1WL 44247815 EC50 = 630.96 nM T59679 C84OVA 44247941 EC50 = 5.012 nM T59679 CA0Q1Z 44247943 EC50 = 3.162 nM T59679 C8EGA3 44247945 EC50 = 1584.89 nM T59679 C0NG8P 44247947 EC50 = 398.11 nM T59679 CS09ZV 44247949 EC50 = 1000 nM T59679 CS5TZ2 44247953 EC50 = 0.631 nM T59679 C9FNH0 44248066 EC50 = 19.95 nM T59679 CA2LC9 44248068 EC50 = 12.59 nM T59679 CK3W2F 44248070 Ki = 15.85 nM T59679 CT40GA 44248072 EC50 = 15.85 nM T59679 CQ9FL7 44248076 EC50 = 1.585 nM T59679 C2B6LX 44248184 EC50 = 1.259 nM T59679 CXE3V4 44248186 EC50 = 0.7943 nM T59679 CDR3G2 44248191 EC50 = 2.512 nM T59679 C0GEP2 44248193 EC50 = 3.162 nM T59679 CEFQ24 44248195 EC50 = 2.512 nM T59679 CU94FE 44248310 EC50 = 79.43 nM T59679 CP2D6Z 44248315 Ki = 1.995 nM T59679 C5DL4T 44248317 EC50 = 10 nM T59679 CL78VT 44248319 EC50 = 0.631 nM T59679 CE19PL 44248321 EC50 = 0.7943 nM T59679 CNI3D4 44248435 EC50 = 1 nM T59679 C64KPA 44248437 Ki = 3.981 nM T59679 C6DJA0 44248439 EC50 = 1.995 nM T59679 C79RLP 44248679 EC50 = 2.512 nM T59679 CDH96L 44248680 EC50 = 1 nM T59679 CW15ZD 44248794 EC50 = 316.23 nM T59679 CLR7B6 44248795 Ki = 3981.07 nM T59679 CTG74J 44248796 Ki = 316.23 nM T59679 CYTC98 44248797 EC50 = 25.12 nM T59679 C13CPM 44248921 EC50 = 0.7943 nM T59679 C38OES 44248922 EC50 = 0.631 nM T59679 C0XK2W 44248923 EC50 = 1.259 nM T59679 C4AML5 44248925 EC50 = 5.012 nM T59679 CZ8M4R 44249053 EC50 = 100 nM T59679 C8DFW0 44249179 EC50 = 501.19 nM T59679 CP2DJ9 44249183 EC50 = 3.162 nM T59679 CQ82PZ 44249186 EC50 = 100 nM T59679 C4KFL7 44249188 EC50 = 15.85 nM T59679 CL0U1W 44249311 EC50 = 158.49 nM T59679 C8MYN0 44249315 EC50 = 7.943 nM T59679 C2L0CK 44249318 Ki = 3162.28 nM T59679 CUXH48 44352308 Ki = 380 nM T59679 CHVO12 44390192 Ki = 0.1995 nM T59679 CI5B1L 44390214 Ki = 0.1259 nM T59679 C2DG5I 44390227 Ki = 0.2512 nM T59679 CD58AW 44390243 Ki = 0.1585 nM T59679 C4Q5IH 44390250 Ki = 0.3162 nM T59679 CD41YC 44390256 Ki = 0.02512 nM T59679 CO4Z6V 44404955 Ki = 6 nM T59679 CZL01O 44404958 Ki = 7 nM T59679 COF9L1 44404960 Ki = 5 nM T59679 CRJD14 44404961 Ki = 9 nM T59679 C64FWU 44404962 Ki = 16 nM T59679 CGK5L0 44404964 Ki = 13 nM T59679 CS29XU 44404965 Ki = 5 nM T59679 C9LEY5 44404966 Ki = 8 nM T59679 CZ9P3U 44404968 Ki = 14 nM T59679 CJ18ER 44404969 Ki = 47 nM T59679 C3SA5V 44427806 Ki = 15 nM T59679 C12XGE 44456400 Ki > 10000 nM T59679 CU52SI 44461665 EC50 = 125.89 nM T59679 CO2P6W 44582815 EC50 = 4 nM T59679 CFSB52 44592414 Ki = 1.413 nM T59679 CNR3K1 44626294 EC50 = 90 nM T59679 C5ABG6 44626295 EC50 = 120 nM T59679 C7NIU3 44628133 Ki = 5.012 nM T59679 CE6M8G 44628198 Ki = 1.995 nM T59679 CERD02 44628200 Ki = 1.995 nM T59679 CIM8C4 44628201 Ki = 10 nM T59679 C2EW5K 44628269 Ki = 199.53 nM T59679 CR4UX9 44629279 Ki = 1.995 nM T59679 C4AEZ5 44629280 Ki = 7.943 nM T59679 CAGF30 44629348 Ki = 125.89 nM T59679 C1XQ8G 44629350 Ki = 2.512 nM T59679 CT0Y4W 45485562 IC50 > 10000 nM T59679 CE9D2C 45485563 IC50 = 5000 nM T59679 CSML06 45485564 IC50 > 10000 nM T59679 CQU3S9 45485604 IC50 > 10000 nM T59679 CG5QJ0 45485614 IC50 > 10000 nM T59679 CE4ZG1 45485619 IC50 > 10000 nM T59679 CSK1X6 45485620 IC50 = 6100 nM T59679 CCY98N 45485624 IC50 > 10000 nM T59679 CREQ49 45485653 IC50 = 4600 nM T59679 CTQ1U3 45485675 IC50 > 10000 nM T59679 C3BC9N 46905984 Ki = 15 nM T59679 C7JB8W 46906000 IC50 > 10000 nM T59679 C83NXB 46935596 Ki = 0.0631 nM T59679 COY21M 46935743 Ki = 0.1259 nM T59679 CVX35K 49780155 Ki = 7.8 nM T59679 CX48MJ 49783206 Ki = 33 nM T59679 CZN2U8 49783207 EC50 = 8.913 nM T59679 C0OT7D 49783208 Ki = 6.3 nM T59679 C2LZJ0 49783209 Ki = 2 nM T59679 CH6P9L 49783210 Ki = 4.5 nM T59679 CW5XT7 49783211 Ki = 7.4 nM T59679 CELG02 49783212 EC50 = 15.85 nM T59679 CG6B3H 49783414 EC50 = 0.1778 nM T59679 C57SMG 49783415 Ki = 2.4 nM T59679 CSK2C4 49783416 Ki = 8664 nM T59679 CI3WS0 49783417 Ki = 17 nM T59679 CXRZ62 49783418 Ki = 12 nM T59679 C0TG6I 49783419 Ki = 2.1 nM T59679 C0TNF2 49783420 Ki = 17 nM T59679 C7ONP3 49783421 Ki = 11 nM T59679 CR40BA 49836386 IC50 > 30000 nM T59679 C0M5XC 49836496 IC50 > 30000 nM T59679 CW42KH 50898699 Ki = 0.06457 nM T59679 CUS21E 50898775 Ki = 0.1413 nM T59679 CL4U8G 50898776 Ki = 0.0537 nM T59679 C1W6TV 50898777 Ki = 0.1072 nM T59679 CXMZ73 50898778 Ki = 1.549 nM T59679 CX48AD 51002362 EC50 > 10000 nM T59679 CM4XO6 52941718 Ki > 1000 nM T59679 CAZ0O4 52945318 Ki = 1.4 nM T59679 C4UCY5 53317702 Ki = 0.195 nM T59679 CB6P5M 53318013 Ki = 2.455 nM T59679 CLNO04 53318069 Ki = 0.8128 nM T59679 CG4XE7 53318070 Ki = 107.15 nM T59679 C9REN0 53319410 Ki = 0.1023 nM T59679 C5HEB1 53319411 Ki = 0.3388 nM T59679 CF39ZT 53319412 Ki = 0.001445 nM T59679 C92KMO 53320666 Ki = 5.012 nM T59679 COUD85 53320711 Ki = 0.2344 nM T59679 C5Z1DR 53320712 Ki = 1.122 nM T59679 CBO6J5 53320713 Ki = 1.995 nM T59679 CDY0J1 53321958 Ki = 2.042 nM T59679 CE03UV 53322003 Ki = 0.7586 nM T59679 CSVZ38 53322004 Ki = 1.259 nM T59679 CLB3X2 53324017 Ki = 2.818 nM T59679 CW4E5I 53324684 Ki = 0.3388 nM T59679 CL7ZM9 53325605 Ki = 0.04266 nM T59679 CFT23B 53325991 Ki = 3630.78 nM T59679 CN7Q0W 53357011 EC50 = 0.4 nM T59679 C08MVZ 53357016 EC50 = 1.9 nM T59679 CXDP95 53357029 Ki = 0.36 nM T59679 C75PML 54677674 EC50 = 17 nM T59679 CXKD25 66810955 Ki = 0.5012 nM T59679 CK8V6A 67211178 Ki = 398.11 nM T59679 C7V8QD 67251061 Ki = 19.95 nM T59679 C1LEH8 67268994 Ki > 10000 nM T59679 CW6ON4 67276147 EC50 = 12.59 nM T59679 C1BLC2 67276168 EC50 = 7.943 nM T59679 CV75GR 67276466 EC50 = 6.31 nM T59679 CX60UI 67472601 Ki = 2.512 nM T59679 C32GEY 67922794 IC50 = 560 nM T59679 CWE97U 68490431 Ki = 0.7943 nM T59679 C7MB8R 68591735 IC50 = 592 nM T59679 CM5ZS8 68592173 IC50 = 118 nM T59679 C2J0MD 68592299 IC50 = 329 nM T59679 C8YG7Z 68592484 IC50 = 648 nM T59679 C54QNY 68592631 IC50 = 73 nM T59679 C6UW1R 68592632 IC50 = 52 nM T59679 CP29IA 68592826 IC50 = 134 nM T59679 C2GSP7 68593153 IC50 = 78 nM T59679 C2PJN0 68593295 IC50 = 178 nM T59679 C62QGB 68593458 IC50 = 190 nM T59679 C1Q2UZ 68593479 IC50 = 1271 nM T59679 CKQ4O9 68593622 IC50 = 377 nM T59679 CSQY72 68593732 IC50 = 805 nM T59679 C2VIM9 68593774 IC50 = 5759 nM T59679 CE6X8W 68593871 IC50 = 493 nM T59679 C7QPC3 70682173 Ki = 1.995 nM T59679 CO2QI6 70682705 EC50 = 31.62 nM T59679 CJ8N6A 70684288 Ki = 2.512 nM T59679 CLJW12 70684789 Ki = 50.12 nM T59679 CM2VZ0 70684790 EC50 = 10 nM T59679 CEDF90 70686434 EC50 = 0.631 nM T59679 CPDY26 70686942 Ki = 100 nM T59679 CI41ON 70686943 EC50 = 19.95 nM T59679 C6KQM1 70688534 Ki = 3.981 nM T59679 CG5MD7 70688535 Ki = 1.585 nM T59679 CY59JW 70691118 EC50 = 19.95 nM T59679 CGL7X5 70694780 Ki = 0.7943 nM T59679 C75VPI 70695321 EC50 = 5.012 nM T59679 CFU25I 70695322 EC50 = 12.59 nM T59679 CK6DA7 70695323 EC50 = 25.12 nM T59679 C32BML 70696825 Ki = 1 nM T59679 C7CM4Y 70696826 Ki = 1 nM T59679 C7SR5N 71450132 Ki = 0.27 nM T59679 C3XNC2 71450247 Ki = 5 nM T59679 CB96KL 71451951 Ki = 0.74 nM T59679 CYH4T1 71452073 Ki = 403 nM T59679 CAQF34 71455625 Ki = 0.03981 nM T59679 C7MNB5 71457264 EC50 > 10000 nM T59679 CHB5W6 71457299 Ki = 0.5012 nM T59679 CMJ1O9 71457409 Ki = 0.26 nM T59679 CRP65E 71459131 Ki = 31.62 nM T59679 CS83IF 71459269 Ki = 0.23 nM T59679 CF73ME 71460941 Ki = 5.2 nM T59679 CK6TP4 71461048 Ki = 33 nM T59679 C63YLA 71461049 Ki = 17 nM T59679 CJD96I 71461050 Ki = 3.1 nM T59679 C0E4XF 71462650 Ki = 0.97 nM T59679 CG4L3C 71462651 Ki = 0.29 nM T59679 CV7X3F 71462652 EC50 = 1.7 nM T59679 C4P3JU 71462776 Ki = 1.2 nM T59679 C3GUQ2 71462777 Ki = 7.5 nM T59679 CUG93T 71712325 Ki = 1.259 nM T59679 CZ0C2S 71712326 Ki = 0.3162 nM T59679 CJF19S 71712327 Ki = 0.7943 nM T59679 C2HBK3 71712328 Ki = 1.585 nM T59679 CUG29A 71712329 EC50 = 3.162 nM T59679 CZ5B9H 71712463 EC50 = 0.3981 nM T59679 CT2I5Z 71712464 EC50 = 1.995 nM T59679 C4EXG5 71712465 EC50 = 1.585 nM T59679 C98QJG 71712466 Ki = 1 nM T59679 C0RDS6 71712611 Ki = 6.31 nM T59679 C9J8ST 71712612 EC50 = 251.19 nM T59679 CL6RN0 71712613 Ki = 251.19 nM T59679 CIH6T3 71714540 Ki = 0.5012 nM T59679 CJ2SI1 71714541 Ki = 0.5012 nM T59679 CJQ45N 71714542 Ki = 0.5012 nM T59679 C8RO7X 71714543 EC50 = 3.162 nM T59679 CS0YC8 71714544 EC50 = 0.7943 nM T59679 C6EG3T 72697299 Ki = 3.981 nM T59679 CIQ29F 72697441 Ki = 0.631 nM T59679 CN2GV9 72697443 Ki = 0.05012 nM T59679 C78LYM 72698087 Ki = 0.11 nM T59679 C63HPK 72698088 Ki = 0.2 nM T59679 CC6Q5R 72771081 Ki < 100 nM T59679 CT1XL6 73352589 Ki = 0.001259 nM T59679 CKE34S 73354085 Ki = 794.33 nM T59679 C2E7QW 75201901 Ki = 9100 nM T59679 C8IDL3 75306277 Ki > 1000 nM T59679 CXT0N2 76313431 Ki = 63.1 nM T59679 C8SVX3 77105903 EC50 = 0.6 nM T59679 CZ75NQ 86582973 Ki = 6.6 nM T59679 C2EMU3 87509467 IC50 = 155 nM T59679 CH7N2Y 87509988 IC50 = 593 nM T59679 CLF6E9 90644470 IC50 = 203 nM T59679 C9TEL6 90644472 IC50 = 916 nM T59679 C63LKR 90644473 IC50 = 110 nM T59679 CCQY39 90644474 IC50 = 195 nM T59679 CYD78E 90644475 IC50 = 453 nM T59679 CQ2MP0 90666907 IC50 = 1.4 nM T59679 C76AKI 91754444 Ki = 0.07943 nM T59679 C7HOY0 118712567 Ki = 501.19 nM T59679 CP85NJ 118712568 Ki = 1000 nM T59679 CHER53 118712569 Ki = 0.1995 nM T59679 CM14CG 118712570 Ki = 1 nM T59679 CUNE23 118712571 Ki = 0.05012 nM T59679 C6X9AQ 118712572 Ki = 0.1995 nM T59679 CZ1CV2 118712573 Ki = 0.1995 nM T59679 CN3D5B 118712574 Ki = 0.2512 nM T59679 CZ0E3N 118712575 Ki = 0.1995 nM T59679 COQ18W 118712576 Ki = 1.259 nM T59679 C8RP6X 118712577 Ki = 1.585 nM T59679 C5A4XS 118712578 Ki = 1.259 nM T59679 CD1L4H 118712579 Ki = 1.259 nM T59679 CP2S6F 118712580 Ki = 0.3162 nM T59679 C4QM2E 124247485 Ki > 10000 nM T59679 C76CNA 127027374 IC50 = 1121 nM T59679 C15EJA 127027375 IC50 = 66 nM T59679 CK8M1R 127027397 IC50 = 1165 nM T59679 C1PZ5S 127027702 IC50 = 954 nM T59679 CJ61PC 127028946 IC50 = 920 nM T59679 CWI3P8 127037816 EC50 > 10000 nM T59679 C8SK3G 127037817 EC50 = 1061 nM T59679 CB41IW 127037818 EC50 = 20 nM T59679 CZU7Q2 127037819 EC50 = 8.7 nM T59679 CDW02Q 127037820 EC50 = 19.8 nM T59679 C5VF7R 127037821 EC50 = 34 nM T59679 C5WN8G 127038354 EC50 = 47 nM T59679 CE63PY 127038726 EC50 = 40 nM T59679 CLN20Q 127039167 EC50 = 10 nM T59679 CA7CD6 127039168 EC50 = 72.3 nM T59679 CR2BC4 127039169 EC50 = 53 nM T59679 CJ51EZ 127039170 EC50 = 840 nM T59679 C3O7CA 127039374 EC50 = 18 nM T59679 C1UN3Y 127039503 EC50 = 520 nM T59679 C1O7YS 127039504 EC50 = 857 nM T59679 CG9BC1 127039505 EC50 = 500 nM T59679 CC40KA 127039506 EC50 = 736 nM T59679 CU74EV 127039507 EC50 = 132 nM T59679 CPWO68 127039508 EC50 = 196 nM T59679 CA4ZB8 127039509 EC50 = 3.9 nM T59679 CI1SB0 127039510 EC50 = 25 nM T59679 C6OBE7 127039819 EC50 = 2247 nM T59679 C9H3EW 127039820 EC50 = 13.2 nM T59679 C8VBS1 127039821 EC50 = 18 nM T59679 C58KTR 127039822 EC50 = 18.3 nM T59679 C8MT7D 127039823 EC50 = 20.7 nM T59679 C20VKF 127039824 EC50 = 31 nM T59679 C1T3UV 127039825 EC50 = 9.7 nM T59679 C7PU6F 127041479 EC50 = 4.8 nM T59679 CSNE69 127041480 EC50 = 11 nM T59679 CF96EA 127041481 EC50 = 9.8 nM T59679 CB2UK6 127041779 EC50 = 633 nM T59679 C04VGO 127041780 EC50 = 1358 nM T59679 C4UE3N 127041781 EC50 = 315.7 nM T59679 CK3CD1 127041782 EC50 = 56.7 nM T59679 C6HB0F 127041783 EC50 = 3.4 nM T59679 C7L9GZ 127041784 EC50 = 15.5 nM T59679 C9HG0Y 127041785 EC50 = 50 nM T59679 CQ1U5D 127041786 EC50 = 49 nM T59679 CFG9O0 127042083 EC50 = 144 nM T59679 C63OPL 127042084 EC50 = 40 nM T59679 CAP82F 127042085 EC50 = 49 nM T59679 CUQL57 127042086 EC50 = 144 nM T59679 CS29LZ 127042087 EC50 = 467 nM T59679 CT4YF8 127042088 EC50 = 88 nM T59679 CUSV58 127042089 EC50 = 39 nM T59679 C70BNG 127042090 EC50 > 10000 nM T59679 C4O1GD 127042670 EC50 = 5.7 nM T59679 C50GOC 130442480 Ki > 10000 nM T59679 CM04RF 130442572 Ki > 10000 nM T59679 CZQS20 134828069 Ki = 150 nM T59679 CYB5V2 134828071 Ki = 40.9 nM T59679 C6N8GM 135367405 Ki > 10000 nM T59679 C6LU0C 135367816 Ki > 10000 nM T59679 CD2TH9 135367820 Ki > 10000 nM T59679 C5AMD9 135367857 Ki > 10000 nM T59679 CV4E6W 136118635 Ki = 2359 nM T59679 CYS3M8 136118637 Ki = 2214 nM T59679 C0UH1B 136118638 Ki = 1063 nM T59679 C6G4AY 136118639 Ki = 3799 nM T59679 C40VES 136118640 Ki = 5308 nM T59679 CH4Q8O 136118646 Ki = 2345 nM T59679 C43JTG 136118647 Ki = 928 nM T59679 CLH0V9 136118648 Ki = 472 nM T59679 C76XEJ 136118649 Ki = 226 nM T59679 CN0V5C 136118650 Ki = 1156 nM T59679 CR72MQ 136118651 Ki = 603 nM T59679 CMP8U3 138376515 EC50 = 6 nM T59679 C9P6BL 145963829 EC50 > 10000 nM T59679 CT0LC2 145964080 EC50 = 42 nM T59679 CHDN35 145964150 IC50 > 10000 nM T59679 CXE7D5 145964157 EC50 = 8.7 nM T59679 CJ26EY 145964746 EC50 = 79 nM T59679 CQ2A9E 145964870 EC50 = 17 nM T59679 CHG3V4 145965246 EC50 = 0.4 nM T59679 CUW2P5 145965547 EC50 > 10000 nM T59679 C6UTC9 145965914 EC50 = 8.4 nM T59679 CXN43I 145966095 EC50 > 10000 nM T59679 C6SJ3Q 145966243 EC50 = 598 nM T59679 C0DWP8 145966407 EC50 = 10.4 nM T59679 CUN21P 145966863 EC50 = 7.3 nM T59679 C86RLP 145967487 EC50 = 0.6 nM T59679 CFV7L2 145968234 EC50 = 687 nM T59679 CJPH53 145968730 EC50 = 9 nM T59679 CD69HW 145972323 EC50 = 36 nM T59679 C86TFR 145972565 EC50 > 10000 nM T59679 CU13IP 145972573 EC50 = 6 nM T59679 CM6BC0 145972577 EC50 = 0.7 nM T59679 C0IA9K 145973097 EC50 = 0.3 nM T59679 C7NGV5 145973678 EC50 > 10000 nM T59679 CFE41Q 145973928 EC50 = 0.1 nM T59679 CPM8Y1 145973946 EC50 = 13.6 nM T59679 CA56TF 145974160 EC50 = 98 nM T59679 CN1UX0 145974756 EC50 = 291 nM T59679 CL1BY7 145975035 EC50 = 1.5 nM T59679 CL2UK4 145975067 EC50 = 4.9 nM T59679 CT8C2M 145975076 EC50 = 34.2 nM T59679 C6EJK7 145975193 EC50 = 0.3 nM T59679 C34KLT 145975297 EC50 = 54 nM T59679 C5NEG9 145975740 EC50 = 114 nM T59679 C71CYU 145975946 IC50 > 10000 nM T59679 CEC8J0 145976249 EC50 = 1941 nM T59679 C54MXJ 145977034 EC50 = 8.8 nM T59679 COAB81 145977126 EC50 = 1941 nM T59679 CELO30 145977409 EC50 = 796 nM T59679 C8RGF2 145977443 EC50 = 48 nM T59679 CEB1M8 145977971 EC50 = 1090 nM T59679 C8RNM6 145978067 EC50 = 8.4 nM T59679 CKF0H6 145978151 EC50 = 758 nM T59679 CFC5J9 145978459 EC50 = 13.8 nM T59679 C86AKO 145978541 EC50 = 65 nM T59679 C9ZL1N 145978825 EC50 = 484 nM T59679 CC2G1V 146025727 Ki = 3700 nM T59679 C0LR8C 155517675 Ki = 37.5 nM T59679 C5D2CI 155523661 Ki = 51 nM T59679 C2K8PD 155525723 EC50 = 4.5 nM T59679 C3XW6I 155543353 EC50 = 2.8 nM T59679 CE32TS 155544687 Ki = 49.6 nM T59679 C8KG6D 155545651 Ki = 37.5 nM T59679 CHT84O 155554403 EC50 = 360 nM T59679 C4GD7W 155558212 EC50 = 72 nM T59679 CV7M0E 155559813 Ki = 25 nM T59679 CY32KD 155565664 EC50 = 1.4 nM T59679 CS7UD8 10574402 EC50 = 25.12 nM T59679 C7CLW1 10757502 EC50 = 39.81 nM T59679 CQ5N3J 10837280 EC50 = 10 nM T59679 COT2U5 15231247 EC50 = 100 nM T59679 CN9JP1 44247817 EC50 = 12.59 nM T59679 CZ45TX 44247820 EC50 = 1.259 nM T59679 C4Y2JB 44247822 EC50 = 1.259 nM T59679 CBKS58 44247951 EC50 = 1.259 nM T59679 C06PRI 44248080 EC50 = 3.981 nM T59679 CMK26V 44248187 EC50 = 39.81 nM T59679 CAU2C3 44248189 EC50 = 0.3981 nM T59679 C03SUN 44248311 Ki = 31.62 nM T59679 C38PDE 44248312 EC50 = 19.95 nM T59679 C05ARK 44248313 EC50 = 1 nM T59679 CX9G1W 44248433 EC50 = 6.31 nM T59679 C68TZP 44248434 EC50 = 3.162 nM T59679 C4WYF7 44248552 Ki = 15.85 nM T59679 CHCF30 44248793 EC50 = 12.59 nM T59679 CAJ83G 44249055 EC50 = 31.62 nM T59679 CR73FT 44249056 EC50 = 39.81 nM T59679 C5WQV1 44249057 EC50 = 15.85 nM T59679 C13PIS 44249189 EC50 = 6.31 nM T59679 CI90JM 44249316 EC50 = 15.85 nM T59679 C3H1SZ 44249317 EC50 = 2511.89 nM T59679 D00OBS 44559159 Ki > 10000 nM T59679 D00PCE 9797313 EC50 = 72.44 nM T59679 D01KAX 135453290 Ki = 515 nM T59679 D03DET 10287730 Ki < 5011.87 nM T59679 D04AQE 1833 Ki = 26.92 nM T59679 D04AZE 3277600 Ki < 10000 nM T59679 D05XGR 6918647 Ki = 2511.89 nM T59679 D05ZUX 44207909 Ki >= 1000 nM T59679 D06HYB 5311299 Ki = 1 nM T59679 D07LRJ 5312149 Ki = 3981.07 nM T59679 D07OSA 133076 EC50 = 2.512 nM T59679 D08CKM 9863250 Ki < 10000 nM T59679 D08JLW 119376 Ki = 0.03981 nM T59679 D08OFG 11177588 Ki = 1910 nM T59679 D09HJL 10331436 Ki = 1700 nM T59679 D09WIL 10028436 Ki = 1905.46 nM T59679 D0AK9V 23673468 Ki = 36 nM T59679 D0B5MU 5311423 Ki = 2.2 nM T59679 D0F6CD 5202 EC50 = 12 nM T59679 D0FE7A 183782 EC50 = 2 nM T59679 D0H7PC 6918553 Ki > 5011.87 nM T59679 D0O3PE 44391713 Ki = 0.7943 nM T59679 D0T2RY 9948320 Ki >= 1000 nM T59679 D0W8EP 5191 Ki = 6.31 nM T82262 D0E3TC 44259 IC50 = 33.6 nM T82262 D0PO8N 117881270 IC50 = 680 nM T82262 CA47TS 3546 Ki = 13000 nM T82262 C0W4UD 3896 IC50 = 200 nM T82262 C18WEB 490561 Ki = 1.8 nM T82262 CM15LD 11521534 IC50 = 398.11 nM T82262 CE5H7D 11544170 IC50 = 199.53 nM T82262 C38FDZ 16760660 IC50 = 10 nM T82262 CI1TV2 44529801 IC50 = 125.89 nM T82262 C3VRO9 44557921 IC50 > 10000 nM T82262 COFN91 45268287 IC50 = 1258.93 nM T82262 CH4B1K 45270042 IC50 = 25.12 nM T82262 CSEA01 45271705 IC50 = 19.95 nM T82262 C47DGZ 59812076 IC50 = 50.12 nM T82262 CV63UL 67240318 IC50 > 10000 nM T82262 CIJ9E2 68778271 IC50 = 3.981 nM T82262 CS1V9U 68778433 IC50 = 50.12 nM T82262 CX75YR 73352604 IC50 = 199.53 nM T82262 C9WJ4H 101510163 IC50 = 40400 nM T82262 COG2M5 136242661 Ki = 15 nM T82262 C04YDK 137248544 Ki = 31 nM T82262 CMB78I 137301774 Ki = 85 nM T82262 CI1E8V 137634241 IC50 = 1910 nM T82262 C6L3HN 137634634 IC50 = 53 nM T82262 CW3RV1 145953992 IC50 = 12.59 nM T82262 CCL34O 145954234 IC50 = 1.585 nM T82262 C4ZH8E 145954241 IC50 = 19.95 nM T82262 CNT8O5 145954713 IC50 = 31.62 nM T82262 CB0F7N 145955167 IC50 = 15.85 nM T82262 C5F4HK 145955417 IC50 = 1995.26 nM T82262 CZ08MB 145960580 IC50 = 31.62 nM T82262 CJDG56 145960632 IC50 = 251.19 nM T82262 CB7TW3 145960672 IC50 = 12.59 nM T82262 CH6G1S 145960935 IC50 = 12.59 nM T82262 C6ZJQ4 145961055 IC50 = 12.59 nM T82262 CZO6T7 145961089 IC50 = 1584.89 nM T82262 CP4JQ5 145961101 IC50 = 3981.07 nM T82262 CX6T3J 145961172 IC50 = 19.95 nM T82262 C54ZQA 145961234 IC50 = 1584.89 nM T82262 C83FPK 145961240 IC50 = 25.12 nM T82262 C9Y8QN 145961342 IC50 = 125.89 nM T82262 C31QBE 145961348 IC50 = 1258.93 nM T82262 CE21QP 145961382 IC50 = 398.11 nM T82262 CWQ27R 145961386 IC50 = 2511.89 nM T82262 CB6S8E 145961504 IC50 = 1584.89 nM T82262 CQ9FN7 145961544 IC50 = 1.995 nM T82262 COCG81 145961565 IC50 = 7.943 nM T82262 C73MVW 145961583 IC50 = 1.995 nM T82262 C23GXR 145961663 IC50 = 25.12 nM T82262 CH40GS 145961699 IC50 = 3981.07 nM T82262 CYLV69 145961794 IC50 = 794.33 nM T82262 C6HB9M 145961899 IC50 = 1584.89 nM T82262 CJ0K8Z 145962062 IC50 = 25.12 nM T82262 CYB36S 145962151 IC50 >= 10000 nM T82262 CV0T1U 145962184 IC50 = 12.59 nM T82262 C6KJG2 145962321 IC50 = 199.53 nM T82262 CJ7NZ0 145962508 IC50 >= 10000 nM T82262 CA2RO4 145962531 IC50 = 7.943 nM T82262 CRQ18V 145962662 IC50 = 398.11 nM T82262 C0UQE1 145962754 IC50 = 1995.26 nM T82262 CCL79I 145963000 IC50 = 12.59 nM T82262 CLFQ85 145963006 IC50 = 100 nM T82262 C0YGB7 145963091 IC50 >= 10000 nM T82262 CG6H2Q 145963149 IC50 >= 10000 nM T82262 CI0V8W 145963248 IC50 = 6.31 nM T82262 CYZ14S 145963250 IC50 = 251.19 nM T82262 CAD5Q9 145963302 IC50 = 501.19 nM T82262 C0JX1P 145963398 IC50 = 15.85 nM T82262 C35ZRP 145963416 IC50 = 316.23 nM T82262 C9CKB4 145963516 IC50 = 100 nM T82262 CJZ4G3 145963549 IC50 = 31.62 nM T82262 CT5XD0 145963609 IC50 = 15.85 nM T82262 CP20IG 145963628 IC50 = 199.53 nM T82262 CC06NJ 145963643 IC50 = 630.96 nM T82262 C9V6AQ 145963687 IC50 = 19.95 nM T82262 C72FZS 145963722 IC50 = 1584.89 nM T82262 C2MD1Q 155513187 IC50 > 10000 nM T82262 D01MNK 25125014 IC50 = 2450 nM T82262 D09FFE 449241 Ki = 29700 nM T82262 D0F3FC 25022668 IC50 = 7.943 nM T17656 D0E3TC 44259 IC50 = 204 nM T17656 D0AV6X 25160990 IC50 > 20000 nM T17656 CR5F4X 6195 IC50 > 20000 nM T17656 C12TIO 6998 IC50 > 20000 nM T17656 C9LD6W 7024 IC50 > 20000 nM T17656 C3ET2I 12819 IC50 = 9732 nM T17656 CV3O5S 16790 IC50 > 20000 nM T17656 CITN94 79352 IC50 > 20000 nM T17656 CHT53C 113099 IC50 > 20000 nM T17656 CD8J9V 11963346 IC50 > 50000 nM T17656 CMGU60 12934390 IC50 = 206 nM T17656 CB1MY8 60196244 IC50 = 290 nM T17656 CRX81Q 71575642 IC50 > 10000 nM T17656 CLTG58 78350466 IC50 = 14 nM T17656 C31OAQ 86290367 IC50 = 472 nM T17656 CLY3D1 86290407 IC50 = 296 nM T17656 CG6YQ8 86290408 IC50 = 181 nM T17656 CU1R5A 86290409 IC50 = 118 nM T17656 C0V5OB 86290410 IC50 = 111 nM T17656 C1VBT9 86290411 IC50 = 118 nM T17656 C8EXO1 86290412 IC50 = 150 nM T17656 CS75OW 86290413 IC50 > 20000 nM T17656 CO84KL 86290454 IC50 > 20000 nM T17656 CY2TV9 86290455 IC50 = 3051 nM T17656 CX32CK 86290456 IC50 > 20000 nM T17656 CP6M9F 86290457 IC50 > 20000 nM T17656 CXK21B 86290458 IC50 = 1230 nM T17656 CT4L8U 86290459 IC50 = 113 nM T17656 CGKV34 86290460 IC50 = 303 nM T17656 CE24CR 86290499 IC50 = 255 nM T17656 CS15PM 86290501 IC50 > 20000 nM T17656 C3V8DA 86290502 IC50 > 20000 nM T17656 C7CTJ6 86290503 IC50 > 20000 nM T17656 CJ81IB 86290504 IC50 = 1718 nM T17656 CUIK08 86290505 IC50 = 4109 nM T17656 CD16CO 86290541 IC50 = 5644 nM T17656 CWZ01E 86290542 IC50 > 20000 nM T17656 C17RVZ 86290569 IC50 = 200 nM T17656 CF47RW 86298445 IC50 = 312 nM T17656 CX4H6I 86583042 IC50 > 50000 nM T17656 CGAR65 90656471 IC50 > 20000 nM T17656 CE7TJ5 90656472 IC50 = 16210 nM T17656 CJ2NI1 118721229 IC50 = 71 nM T17656 CC05EY 118721230 IC50 = 14 nM T17656 C7HJ8Y 118721231 IC50 > 99000 nM T17656 C5XMF8 118721232 IC50 = 170 nM T17656 CZY01I 118721233 IC50 = 29 nM T17656 C2USQ7 118721234 IC50 = 51 nM T17656 CDS2U3 118721235 IC50 = 9.7 nM T17656 C0H9OV 118721236 IC50 = 11 nM T17656 C83KJY 118721237 IC50 = 6.4 nM T17656 C13QEP 118721238 IC50 = 5.1 nM T17656 CVC3B0 118721239 IC50 = 14 nM T17656 C2F6MN 118721240 IC50 = 45 nM T17656 C36PRN 118721241 IC50 = 54 nM T17656 CY0J8A 118721242 IC50 = 12 nM T17656 CJLX62 118721243 IC50 = 22 nM T17656 C14BFC 118721244 IC50 = 13 nM T17656 C6ETU2 118721245 IC50 = 31 nM T17656 C4TXF2 118730409 IC50 > 50000 nM T17656 C4X7SD 122192466 IC50 > 10000 nM T17656 CY28AI 135398515 IC50 = 9939 nM T17656 CKO83Y 136664429 EC50 = 143 nM T17656 CPC5O0 137333978 IC50 = 303 nM T17656 CA93HF 139593294 IC50 = 160 nM T17656 C2MD1Q 155513187 IC50 > 10000 nM T17656 CN47JC 155517517 IC50 = 72 nM T17656 C5U0SQ 155521969 IC50 = 130 nM T17656 C8N4OH 155522759 IC50 = 90 nM T17656 CRJF80 155525584 IC50 > 10000 nM T17656 CR51DL 155530872 IC50 > 10000 nM T17656 CN0PW5 155533307 IC50 = 190 nM T17656 CET2Q5 155539312 IC50 = 4060 nM T17656 C1TOM0 155540070 IC50 = 200 nM T17656 C1UM3W 155540082 IC50 = 100 nM T17656 C0RWS7 155542155 IC50 > 10000 nM T17656 CV6ZI7 155543519 IC50 > 10000 nM T17656 C5MHX7 155546098 IC50 = 130 nM T17656 CW4QJ2 155547079 IC50 = 110 nM T17656 CTZ5N8 155548986 IC50 = 160 nM T17656 CIR6U2 155551979 IC50 = 33 nM T17656 CY4P0U 155554101 IC50 = 890 nM T17656 CQH9K8 155555756 IC50 > 10000 nM T17656 CS5OW0 155560180 IC50 = 240 nM T17656 CFOP01 155560487 IC50 = 160 nM T17656 CE5W2A 155560538 IC50 = 2700 nM T17656 C8F6IT 155566735 IC50 = 840 nM T17656 D0E3CB 86290500 IC50 = 47 nM T17656 D0W1NH 72881 IC50 > 20000 nM T81830 D0E3TC 44259 IC50 = 1.24 nM T81830 C3VRO9 44557921 IC50 > 10000 nM T81830 CV63UL 67240318 IC50 > 10000 nM T81830 C5N1VZ 102581295 IC50 > 10000 nM T81830 CGBZ13 134843302 IC50 > 10000 nM T81830 C3MK9W 136807986 IC50 > 10000 nM T81830 C2MD1Q 155513187 IC50 > 10000 nM T81830 C68GMW 155538446 IC50 > 10000 nM T81830 CY6Q8S 155554337 IC50 > 10000 nM T81830 CO2I4P 155559898 IC50 = 1200 nM T99204 CTF47W 25164607 IC50 = 1 nM T99204 CTB5M4 25164609 IC50 = 2 nM T99204 CEKW51 25164812 IC50 = 3 nM T99204 CWX1L8 58445338 IC50 = 8 nM T99204 C8K7BT 71453301 IC50 = 6 nM T99204 C61FYG 71460487 IC50 = 16 nM T99204 C5Y1GS 71462196 IC50 = 20 nM T00863 D0X5SD 3117 IC50 = 320 nM T00863 C49BCY 1570 IC50 = 33000 nM T00863 CZ7IA3 1647 IC50 = 550 nM T00863 CKC31Q 86633 IC50 = 2600 nM T00863 C4ZB8R 245718 IC50 = 75000 nM T00863 C39MKT 712750 IC50 = 35000 nM T00863 COB3T1 2132963 IC50 = 5000 nM T00863 CF2N8O 2794167 IC50 = 5910 nM T00863 C94LDM 6459851 IC50 = 91000 nM T00863 C62ZIW 10176672 IC50 = 30000 nM T00863 C9C6LU 10334080 IC50 = 100000 nM T00863 CCUJ60 10445232 IC50 > 1000000 nM T00863 CY41LT 10445774 IC50 > 1000000 nM T00863 CPIV30 13194096 IC50 > 100000 nM T00863 CW1FA3 16227983 IC50 = 16000 nM T00863 CBZP95 16780874 IC50 = 34000 nM T00863 CMO3B7 29130197 IC50 > 100000 nM T00863 CC9VJ0 39047495 IC50 = 50000 nM T00863 CO6A3U 44387955 IC50 = 100000 nM T00863 C3PTZ7 70700688 IC50 = 54000 nM T00863 C3UBY0 122163387 IC50 = 8700 nM T00863 C4P9JW 122516179 IC50 = 2800 nM T00863 CYT3P6 122516185 IC50 = 7300 nM T00863 CMB23H 122516211 IC50 = 3100 nM T00863 CV25IT 122516222 IC50 = 2900 nM T00863 CU9N2M 122516246 IC50 = 5500 nM T00863 CN3VC8 122516255 IC50 = 2400 nM T00863 C4M3ZK 122516295 IC50 = 3100 nM T00863 C4ELG0 122516336 IC50 = 1800 nM T00863 C9BL6C 122516346 IC50 = 8400 nM T00863 CX3B4R 122516830 IC50 = 83000 nM T00863 C41DZW 122516838 IC50 = 93000 nM T00863 COK0J3 122516959 IC50 = 11000 nM T00863 C0AQW4 122517020 IC50 > 100000 nM T00863 CL3Q9Z 122517043 IC50 = 18000 nM T00863 C84UJE 130302628 IC50 = 1260 nM T00863 CL74FP 132253032 IC50 = 30000 nM T00863 CSEW98 132253084 IC50 = 35000 nM T00863 CG6KP2 132253106 IC50 = 21000 nM T00863 CCL91Y 132253144 IC50 = 23000 nM T00863 C4C6HK 132253151 IC50 = 22000 nM T00863 CJAN-32 132253163 IC50 = 16000 nM T00863 CC89LI 132253175 IC50 = 11000 nM T00863 CS0LC7 134280641 IC50 = 16000 nM T00863 CGN6E7 135492608 IC50 = 9200 nM T00863 CC35GR 135615984 IC50 = 1600 nM T00863 CE9O8V 137634616 IC50 = 45000 nM T00863 CI1Y2F 137648233 IC50 = 3500 nM T00863 CTA4O6 137656044 IC50 = 52000 nM T00863 D02UVS 5455 IC50 = 1040 nM T40192 D04VIS 5318517 IC50 = 49600 nM T40192 D00VUI 6199 IC50 = 3000 nM T40192 CT6YF0 5100 EC50 = 50000 nM T40192 C5SRE2 10658 IC50 = 2500 nM T40192 C2RK6G 16763 IC50 = 110000 nM T40192 CNM70A 16766 IC50 = 28600 nM T40192 CTF38D 16884 IC50 > 300000 nM T40192 C9OQD3 360404 EC50 = 30000 nM T40192 C5OMZ6 372837 IC50 = 119000 nM T40192 C5TE8O 768151 IC50 = 19000 nM T40192 CWZ91D 779509 IC50 = 35200 nM T40192 C1DRF6 906649 EC50 = 6000000 nM T40192 C18YXT 907191 EC50 = 800000 nM T40192 C57UCN 907294 EC50 = 800000 nM T40192 C3KVN0 1609902 IC50 = 60000 nM T40192 CQ84UY 1765149 IC50 = 20000 nM T40192 CX18TZ 1767434 EC50 = 600000 nM T40192 CCT7O6 1910342 IC50 = 20000 nM T40192 CW3XV4 2780275 IC50 = 500 nM T40192 CU8DA2 2780311 IC50 > 10000 nM T40192 C73ZCI 3121122 IC50 = 74400 nM T40192 C7EFX9 3336826 EC50 = 600000 nM T40192 CU6VG2 3377704 EC50 = 60000 nM T40192 CCK3V1 3636895 EC50 = 100000 nM T40192 CQF58I 3729894 EC50 = 600000 nM T40192 CF5MD8 3742469 EC50 = 1000000 nM T40192 CS7C5K 3761756 EC50 = 100000 nM T40192 CA06GK 3840300 EC50 = 80000 nM T40192 C3RV9N 4616261 EC50 = 1000000 nM T40192 CY47VC 4914300 EC50 = 800000 nM T40192 CNZ73E 5280567 IC50 = 200000 nM T40192 CQ8B9L 5387296 EC50 = 50000 nM T40192 CY0CO2 5495925 IC50 = 7500 nM T40192 CE5PN8 7567955 IC50 = 30000 nM T40192 C6DBO0 9910975 IC50 = 50 nM T40192 CU36GT 10342859 IC50 > 10000 nM T40192 C8HO6F 10528296 IC50 > 10000 nM T40192 C5HIV4 10549239 IC50 = 900 nM T40192 C42RZM 10568837 IC50 > 10000 nM T40192 C1JEG0 10595299 IC50 = 380 nM T40192 C3ABP7 10596208 IC50 = 2300 nM T40192 C5ODG9 10598884 IC50 > 10000 nM T40192 CBRV16 10621642 IC50 = 5000 nM T40192 CP4VD3 10623854 IC50 = 2700 nM T40192 C51QFE 10646124 IC50 > 10000 nM T40192 C2SG8N 10667404 IC50 > 10000 nM T40192 C2W6SQ 10672875 IC50 = 1800 nM T40192 CT1MF9 10672927 IC50 = 620 nM T40192 C0EWB4 10674467 IC50 = 4600 nM T40192 C9R5YQ 10695662 IC50 = 170 nM T40192 CWA5X8 10713914 IC50 > 10000 nM T40192 CYCG32 10716340 IC50 > 10000 nM T40192 CUR1B0 10735147 IC50 > 10000 nM T40192 CU97ZN 10736697 IC50 > 10000 nM T40192 C6G1OW 10738057 IC50 = 800 nM T40192 CBNP69 10740754 IC50 = 5000 nM T40192 C2E6DV 10741807 IC50 > 10000 nM T40192 C5NQ1M 10757074 IC50 = 4000 nM T40192 CF01JA 10758135 IC50 = 2300 nM T40192 CGD9B4 10760357 IC50 > 10000 nM T40192 CP89CY 10761093 IC50 = 1200 nM T40192 C39HVX 10768433 IC50 = 1800 nM T40192 CSBY47 10850430 IC50 > 10000 nM T40192 CP9D3N 11797436 IC50 = 280 nM T40192 CO58NY 15698945 IC50 > 10000 nM T40192 C4Q6YN 16462555 IC50 = 40000 nM T40192 C34AUM 21679194 IC50 = 11100 nM T40192 C3VS9X 23606103 EC50 = 4000000 nM T40192 COMI46 23606149 EC50 = 5000000 nM T40192 CL75EX 44226791 IC50 > 10000 nM T40192 C60VSB 46879489 IC50 > 20000 nM T40192 C0SQ2G 46880202 IC50 > 20000 nM T40192 CY89VO 46880203 IC50 > 20000 nM T40192 CHFO19 52941330 IC50 = 5000 nM T40192 CZ65LU 54694372 EC50 = 100000 nM T40192 C8TDR2 71583471 EC50 = 80000 nM T40192 CGTF76 71583472 EC50 = 10000 nM T40192 CB1SF4 71583583 EC50 = 600000 nM T40192 C1YZ6I 71583584 EC50 = 530000 nM T40192 CWU4M2 71583585 EC50 = 60000 nM T40192 CRTN26 71583586 EC50 = 60000 nM T40192 CBY78V 71583587 EC50 = 60000 nM T40192 CS1WR4 71583687 EC50 = 670000 nM T40192 C68AVL 71583688 EC50 = 80000 nM T40192 CBG0V7 71583689 EC50 = 60000 nM T40192 CX90FN 71583803 EC50 = 40000 nM T40192 CV62BU 71583804 EC50 = 40000 nM T40192 C9FI1R 71583805 EC50 = 100000 nM T40192 CGZ39L 71583922 EC50 = 60000 nM T40192 C0BP2Y 71583923 EC50 = 100000 nM T40192 CN2MT4 71583924 EC50 = 10000 nM T40192 C9A2HX 71584028 EC50 = 100000 nM T40192 CWE4U0 71584029 EC50 = 10000 nM T40192 C56HEL 71584030 EC50 = 70000 nM T40192 CR81BG 71584031 EC50 = 100000 nM T40192 C87ISK 71584032 EC50 = 100000 nM T40192 C0I6TR 71584135 EC50 = 60000 nM T40192 CZ0XA9 71584136 EC50 = 700000 nM T40192 C8ZKY0 71584137 EC50 = 600000 nM T40192 C3S2DP 71584138 EC50 = 600000 nM T40192 CU4LH7 71584139 EC50 = 80000 nM T40192 CU0A8Q 71584140 EC50 = 3000000 nM T40192 CK6Y4A 71584253 EC50 = 700000 nM T40192 C1S6LV 71584254 EC50 = 3000000 nM T40192 C1WMO3 71584255 EC50 = 3000000 nM T40192 C4JC5W 71584256 EC50 = 700000 nM T40192 C8R1TD 71584257 EC50 = 700000 nM T40192 CE25MG 71584258 EC50 = 700000 nM T40192 C3OZT8 71584390 EC50 = 3000000 nM T40192 CF8HW3 71584391 EC50 > 10000000 nM T40192 C9A3LS 71584392 EC50 = 3000000 nM T40192 C8LRW4 71584393 EC50 = 1000000 nM T40192 CK5E9W 71584394 EC50 = 1000000 nM T40192 C5W6CX 71584522 EC50 = 700000 nM T40192 D01FEA 392450 IC50 > 20000 nM T40192 D01WTQ 5495929 IC50 > 20000 nM T40192 D04YTE 331783 IC50 = 75 nM T40192 D05WQF 637540 IC50 = 50000 nM T40192 D05YJR 5495926 IC50 > 20000 nM T40192 D06PRC 5281650 IC50 > 20000 nM T40192 D07JDD 46834285 IC50 > 10000 nM T40192 D0J2PO 46887866 IC50 = 2300 nM T40192 D0O8EB 5281633 IC50 > 20000 nM T65570 C8T6GS 13017 Ki = 2300 nM T65570 C6C7ZT 13376 Ki = 7200 nM T65570 CG1I4X 22686 Ki = 5600 nM T65570 CNY4H5 80654 Ki = 31000 nM T65570 CK7LB3 221387 Ki = 5500 nM T65570 CZI0Y4 253317 Ki = 3900 nM T65570 CT83WR 268118 Ki = 22000 nM T65570 C7BCG2 347402 Ki = 3600 nM T65570 C2QIP5 444215 Ki = 2 nM T65570 C6FE8Z 5287890 Ki = 360 nM T65570 C0TYR2 10510948 Ki = 5500 nM T65570 CAQ97C 10535407 Ki = 7400 nM T65570 CJR9A3 10535470 Ki = 1900 nM T65570 CP9N5D 10582973 Ki = 1800 nM T65570 C0XW8H 10583265 Ki = 14000 nM T65570 C2OU9B 10654643 Ki = 5900 nM T65570 CI41XN 10654696 Ki = 24000 nM T65570 CFB7N0 10725554 Ki = 880 nM T65570 C2HM1K 10773209 Ki = 4500 nM T65570 CH9X0P 10773210 Ki = 4500 nM T65570 CG4Y3W 11815987 Ki = 7000 nM T65570 CA0D9M 15475283 Ki = 33000 nM T65570 CUQ1A8 20333386 Ki = 3600 nM T65570 CZ07CP 20336979 Ki = 3800 nM T65570 C0SWI8 44415182 Ki = 400 nM T65570 CY90BD 49818230 IC50 = 460 nM T65570 C8H1CZ 155536201 IC50 = 5600 nM T65570 CMZP19 444170 Ki = 21000 nM T15855 D02EYG 10096344 IC50 > 40000 nM T15855 D0K9MY 11243969 Ki = 130 nM T15855 D0L3DK 6918537 Ki = 810 nM T15855 D0NJ5H 11450633 IC50 > 25000 nM T15855 D0T8XB 44513473 IC50 = 68 nM T15855 D0U2JP 4369359 IC50 = 1820 nM T15855 D04XIO 11253490 IC50 = 8427 nM T15855 D07EPV 11949652 IC50 = 260 nM T15855 D07HZG 11516136 IC50 = 7000 nM T15855 D0FQ2U 6918572 Ki = 1.5 nM T15855 D0M3XR 46209133 IC50 > 67000 nM T15855 D0N6SO 15983988 IC50 > 100000 nM T15855 D04MAZ 71731606 IC50 > 100000 nM T15855 D00FYF 9796290 IC50 = 4573 nM T15855 D0A1NU 16049769 Ki > 30000 nM T15855 D0F3TI 11673176 Ki = 11 nM T15855 D0Q4YP 11996845 IC50 > 100000 nM T15855 CE98OF 6451150 IC50 = 11000 nM T15855 C4RE5F 7020797 IC50 = 115000 nM T15855 CCIX30 9209502 IC50 = 147 nM T15855 C14VRG 9794073 IC50 = 550 nM T15855 CSA6V9 9796352 IC50 = 6600 nM T15855 C7KR1T 9799867 IC50 > 100000 nM T15855 CNJ0Z3 9800721 Ki > 30000 nM T15855 C62DNH 9843297 IC50 = 69000 nM T15855 CZUQ34 9883487 IC50 = 220 nM T15855 C2TV9M 9884543 IC50 = 88 nM T15855 C28XTC 9942425 IC50 > 1000000 nM T15855 CQ8J7T 9953181 IC50 = 62000 nM T15855 CT6XQ2 9983092 IC50 = 8600 nM T15855 C78NMY 10026124 IC50 = 63000 nM T15855 C97FIB 10087948 IC50 > 100000 nM T15855 C83ZDL 10096130 IC50 = 930 nM T15855 C0Q7BK 10127057 IC50 = 75000 nM T15855 C9ERD7 10130575 IC50 = 51 nM T15855 C2H0UF 10149048 Ki = 2 nM T15855 C4CX1P 10157141 IC50 = 46000 nM T15855 C5P0AO 10238227 IC50 = 8000 nM T15855 CZ90LD 10250452 IC50 > 100 nM T15855 CU8C5K 10254918 IC50 > 100000 nM T15855 C17HUN 10255762 IC50 = 70000 nM T15855 C6ER9U 10269517 IC50 = 3400 nM T15855 C3FB4T 10310021 IC50 > 100000 nM T15855 CY6N9I 10318743 IC50 = 55000 nM T15855 CF1S8U 10320144 IC50 > 100000 nM T15855 C08UHI 10320529 IC50 = 8100 nM T15855 CNV4R3 10324641 IC50 = 46000 nM T15855 CM6Y1B 10339570 Ki > 30000 nM T15855 CXP16T 10340933 IC50 = 71000 nM T15855 C1AEN6 10341846 IC50 = 71000 nM T15855 C7UO3L 10376704 Ki > 30000 nM T15855 CQ7J2Z 10383508 IC50 > 20000 nM T15855 CY5M4R 10388027 IC50 = 16000 nM T15855 CHZ85I 10393133 IC50 = 8600 nM T15855 C29MEL 10399628 Ki > 30000 nM T15855 C7R6TZ 10406789 IC50 = 39000 nM T15855 CVK1G5 10412922 IC50 = 7900 nM T15855 C92DAJ 10415172 IC50 = 56000 nM T15855 C1O2RY 10426457 IC50 = 58000 nM T15855 C80ZBS 10429788 IC50 > 100000 nM T15855 C6GHF1 10433039 IC50 = 58000 nM T15855 CWCA76 10439426 IC50 > 100000 nM T15855 CAF71Y 10443207 IC50 = 40500 nM T15855 CO59EL 10450114 IC50 = 46000 nM T15855 C4OC6P 10455620 IC50 = 6000 nM T15855 C1WKE4 10455621 IC50 = 44000 nM T15855 CHP37D 10456407 IC50 > 1000000 nM T15855 CH1DG5 10478099 IC50 = 66000 nM T15855 CK3IW4 10584272 IC50 = 3800 nM T15855 C0KTQ5 10607253 IC50 = 127000 nM T15855 C4PJ7H 10656779 IC50 = 10500 nM T15855 CHA8X6 10751333 IC50 = 26000 nM T15855 CYLO09 10774283 IC50 = 23000 nM T15855 CL26WQ 10780092 IC50 = 242000 nM T15855 C2KDY6 10798619 IC50 = 612000 nM T15855 C1WG0P 10798659 IC50 = 15 nM T15855 C1ZJ4I 10799226 IC50 = 10300 nM T15855 CJKX61 10821833 IC50 = 76000 nM T15855 C7BLJ1 10821834 IC50 > 1000000 nM T15855 C3E8ID 10845163 IC50 = 14000 nM T15855 CK9SB4 10845727 IC50 = 130000 nM T15855 CLA05J 10932707 Ki = 12360 nM T15855 CT75CX 10982631 IC50 > 1000000 nM T15855 C4MD5V 11037154 IC50 > 1000000 nM T15855 CH4TD3 11037548 IC50 > 1000000 nM T15855 C9S8AG 11068388 IC50 = 25000 nM T15855 CA4N0B 11117606 Ki = 1218 nM T15855 CXT8Y2 11151568 IC50 > 100000 nM T15855 C4HBU9 11153488 IC50 > 100000 nM T15855 C7HRW0 11164704 IC50 > 100000 nM T15855 C82GSQ 11165177 IC50 > 100000 nM T15855 C9HKB7 11188314 IC50 > 100000 nM T15855 CF1LD8 11199808 Ki = 538 nM T15855 C68XFD 11205761 IC50 > 1000000 nM T15855 C3BXS4 11206225 IC50 > 1000000 nM T15855 CJB87Z 11210511 IC50 = 21000 nM T15855 CSN6U7 11220682 IC50 = 11000 nM T15855 CU3BG5 11222807 IC50 = 86000 nM T15855 CK1UE7 11229192 IC50 > 500000 nM T15855 CHX25W 11232123 IC50 > 100000 nM T15855 CYL67P 11232890 Ki = 616 nM T15855 CR3PJ9 11233253 IC50 > 100000 nM T15855 C3UA7X 11234761 IC50 > 100000 nM T15855 C32ZGY 11234800 IC50 > 100000 nM T15855 C5AB7G 11236208 IC50 = 19000 nM T15855 CQ6C5F 11246131 IC50 > 100000 nM T15855 C4VQ0N 11246214 IC50 > 100000 nM T15855 C2YS9G 11256520 IC50 > 100000 nM T15855 CKL1A8 11268930 Ki = 155 nM T15855 CM0YI7 11269397 Ki = 191 nM T15855 C5IY0L 11269712 IC50 = 63000 nM T15855 CM1A5F 11270889 IC50 = 5300 nM T15855 CUB62P 11278798 IC50 > 100000 nM T15855 CB5SD1 11280296 IC50 > 100000 nM T15855 CL5SH2 11281817 IC50 = 20000 nM T15855 C1YH5K 11291901 IC50 > 100000 nM T15855 CAW02M 11303089 IC50 > 100000 nM T15855 CDZ79G 11304224 IC50 > 100000 nM T15855 C2SOA8 11306467 IC50 = 80000 nM T15855 C06NLF 11309656 IC50 > 500000 nM T15855 C8I1QE 11310450 IC50 = 139000 nM T15855 C47GSV 11310499 IC50 = 3100 nM T15855 CEZ27P 11314348 Ki = 239 nM T15855 CTG12Q 11321743 IC50 > 500000 nM T15855 CM4CT0 11348315 IC50 > 100000 nM T15855 CNB7G8 11356095 IC50 = 4700 nM T15855 CUH3S7 11360493 IC50 > 100000 nM T15855 CZ93VH 11361944 IC50 = 84000 nM T15855 CKP0G9 11362130 IC50 = 700 nM T15855 CMZ1S9 11373129 IC50 > 100000 nM T15855 C30JEU 11381416 IC50 > 30000 nM T15855 CML13R 11389441 IC50 = 411000 nM T15855 CH35IZ 11392716 IC50 > 100000 nM T15855 CL9HN3 11395030 Ki = 151 nM T15855 CTW02K 11406276 Ki = 241 nM T15855 C9AW7O 11416338 IC50 > 100000 nM T15855 C0RIS4 11417008 IC50 = 58000 nM T15855 C2ZT0L 11418204 IC50 > 100000 nM T15855 CRZ5F1 11418876 IC50 = 69000 nM T15855 CFD62G 11419146 IC50 > 100000 nM T15855 CY15PU 11429829 Ki = 330 nM T15855 CFTC85 11432169 IC50 > 100000 nM T15855 C82ENX 11439333 IC50 > 100000 nM T15855 CRW3G4 11440163 IC50 > 100000 nM T15855 CH09SE 11447824 IC50 = 12500 nM T15855 CZ68MT 11451290 IC50 > 100000 nM T15855 C6US2X 11461807 IC50 = 100000 nM T15855 CV71FH 11464036 IC50 > 100000 nM T15855 CWO06L 11471453 IC50 = 14000 nM T15855 CE5A4M 11475797 IC50 = 12000 nM T15855 C7JWD3 11476287 IC50 = 48000 nM T15855 CS4H7X 11481506 IC50 = 340 nM T15855 C6U9KB 11484559 IC50 > 100000 nM T15855 CTD0S4 11486251 Ki = 2952 nM T15855 CNMA97 11487118 IC50 = 46000 nM T15855 C06RUA 11493219 IC50 > 30000 nM T15855 CDT16S 11493492 Ki > 30000 nM T15855 C9PRY1 11494684 IC50 = 41859 nM T15855 CJD30Y 11495704 IC50 = 53000 nM T15855 CAH5Z6 11500899 IC50 > 30000 nM T15855 CH7VS5 11505454 IC50 = 4300 nM T15855 CM8QB3 11510166 Ki = 13300 nM T15855 CQDM72 11514208 IC50 = 63000 nM T15855 C15UQK 11515912 IC50 = 1407 nM T15855 C0XVU3 11516085 IC50 > 10000 nM T15855 C2S8BH 11516511 Ki > 30000 nM T15855 CH5A7Q 11518007 IC50 = 33000 nM T15855 CJM1L9 11522376 IC50 = 25000 nM T15855 C2TCM8 11523077 IC50 = 1700 nM T15855 C8KB4F 11524437 Ki > 30000 nM T15855 CMYN65 11526865 IC50 > 100000 nM T15855 C0O3XD 11527019 IC50 > 100000 nM T15855 CWH3S0 11529375 IC50 > 100000 nM T15855 COL08I 11529539 IC50 = 32000 nM T15855 CZFI65 11531704 Ki = 5500 nM T15855 C1B8JN 11532057 Ki > 30000 nM T15855 CZ35WN 11533932 IC50 > 100000 nM T15855 COXK41 11537890 Ki > 30000 nM T15855 CKM89Z 11538673 IC50 > 100000 nM T15855 CMD6H8 11538715 IC50 = 1150 nM T15855 CK36XC 11538961 Ki = 5300 nM T15855 CG7I8Z 11538992 IC50 > 100000 nM T15855 CPR71X 11540951 IC50 > 100000 nM T15855 C98GDW 11541277 IC50 > 100000 nM T15855 CBR9K8 11541314 IC50 > 100000 nM T15855 CVT52Y 11545508 IC50 > 100000 nM T15855 C6KBN4 11546261 Ki = 2.4 nM T15855 CJIX61 11547698 IC50 > 10000 nM T15855 CY3RK7 11551987 IC50 > 100000 nM T15855 C2DJ6Y 11552953 Ki > 30000 nM T15855 CA16WP 11554165 IC50 = 30000 nM T15855 C85EQW 11559371 IC50 > 100000 nM T15855 CDK7I5 11559922 Ki = 1.9 nM T15855 CL4D9A 11565911 IC50 = 40000 nM T15855 CMN2K0 11566106 IC50 = 2592 nM T15855 CI5W4Y 11566450 IC50 > 30000 nM T15855 CR37GC 11567606 Ki = 2.2 nM T15855 CY0A7J 11570138 IC50 > 100000 nM T15855 CH76QT 11572962 IC50 > 100000 nM T15855 C6F4OE 11573417 IC50 = 2121 nM T15855 CAE39I 11573427 IC50 > 30000 nM T15855 CCR9Q2 11574031 IC50 = 2387 nM T15855 CE03TL 11574811 Ki > 30000 nM T15855 CQU80H 11576569 IC50 > 100000 nM T15855 CW94NS 11577331 IC50 > 100000 nM T15855 CQ86GI 11577431 IC50 > 100000 nM T15855 CW31KG 11579932 IC50 = 40000 nM T15855 CVG3B6 11580945 IC50 = 21961 nM T15855 CCR0D7 11581247 IC50 = 1700 nM T15855 CYT4Z1 11581458 IC50 > 100000 nM T15855 C9J1NO 11581694 IC50 > 10000 nM T15855 CAZL49 11584650 IC50 > 100000 nM T15855 COH9V8 11589872 IC50 > 10000 nM T15855 C5JYV7 11591936 IC50 > 100000 nM T15855 CSCW37 11592154 IC50 = 28000 nM T15855 CA51WQ 11595401 IC50 = 6300 nM T15855 CO0QJ8 11596007 Ki > 30000 nM T15855 CE8M3K 11596123 Ki > 30000 nM T15855 C9MXO0 11596219 IC50 > 20000 nM T15855 CMUV42 11596607 IC50 = 2390 nM T15855 CSW3M9 11597271 IC50 > 10000 nM T15855 CY4W0X 11602707 IC50 = 4000 nM T15855 CBE6K8 11603637 Ki = 2700 nM T15855 CPXV24 11603996 IC50 > 100000 nM T15855 CL4NM7 11604454 IC50 = 202 nM T15855 C0S2RQ 11605368 IC50 > 10000 nM T15855 C15DLO 11608317 IC50 = 4300 nM T15855 COF62W 11611325 Ki = 3982 nM T15855 CQL5S8 11613750 IC50 > 100000 nM T15855 CZ91WO 11616288 IC50 = 32000 nM T15855 CD3YU1 11616861 IC50 > 30000 nM T15855 CEX4O6 11617338 IC50 = 5346 nM T15855 C2APG7 11623550 IC50 > 30000 nM T15855 CDZ72J 11624893 IC50 > 20000 nM T15855 CRY2D5 11625412 Ki = 7000 nM T15855 C7YKC0 11628195 IC50 > 100000 nM T15855 CV17GF 11631125 IC50 = 50000 nM T15855 CSO1D6 11632159 Ki > 30000 nM T15855 C8Y3FM 11632315 IC50 = 3200 nM T15855 CM1DR9 11632375 Ki > 30000 nM T15855 C09KAV 11632502 IC50 = 8000 nM T15855 CHLA97 11638762 Ki > 30000 nM T15855 CRA0H5 11639131 Ki > 30000 nM T15855 C0M1HR 11640120 IC50 > 10000 nM T15855 C3RZO9 11645337 IC50 = 10744 nM T15855 CQO8U6 11648011 Ki > 30000 nM T15855 CXG1B4 11649741 IC50 > 100000 nM T15855 CZBD50 11653749 Ki > 30000 nM T15855 C94OMG 11654093 Ki > 30000 nM T15855 C8AU5P 11654528 Ki = 3400 nM T15855 C52ION 11655271 Ki > 30000 nM T15855 C43OVS 11673852 IC50 = 20000 nM T15855 CCBS09 11674180 Ki > 30000 nM T15855 CTNO72 11674721 IC50 = 6400 nM T15855 C2G6RP 11675637 Ki = 12200 nM T15855 CI1ED9 11676224 IC50 = 41000 nM T15855 C3Y7EL 11678025 IC50 > 100000 nM T15855 C1A7NS 11680394 IC50 = 80000 nM T15855 CV0XW8 11680991 IC50 = 855.5 nM T15855 CFX6Z9 11681207 IC50 = 32000 nM T15855 CNF1M4 11681778 IC50 > 20000 nM T15855 C0IWC9 11689866 IC50 = 3340 nM T15855 C79ECL 11695535 IC50 = 4169 nM T15855 C7DCV9 11696495 Ki > 30000 nM T15855 C6JPE0 11696912 Ki > 30000 nM T15855 CRU2Q1 11697286 Ki = 1300 nM T15855 C2WK1Z 11697387 Ki = 6800 nM T15855 C8SI4E 11702902 IC50 = 8338 nM T15855 C0Q3IL 11703158 IC50 = 12847 nM T15855 C2X5GC 11704411 Ki = 4700 nM T15855 C6YHK3 11704412 Ki = 7200 nM T15855 CFO63Q 11704578 IC50 = 2117 nM T15855 CU8LZ4 11705859 IC50 = 3416 nM T15855 CZF5D9 11708829 IC50 = 50000 nM T15855 CK4I6J 11710700 Ki > 30000 nM T15855 C04OMI 11711314 Ki > 30000 nM T15855 C8VC2D 11711413 Ki = 6300 nM T15855 C8KD6N 11711414 Ki = 14600 nM T15855 C34BEP 11716483 Ki > 30000 nM T15855 CCR80L 11717090 IC50 = 3583 nM T15855 CZS71R 11717268 IC50 = 5532 nM T15855 C1XD5I 11718004 Ki > 30000 nM T15855 CY1S3Q 11719625 IC50 > 10000 nM T15855 CIEJ54 11720809 IC50 > 100000 nM T15855 CX9U4G 11731880 IC50 > 500000 nM T15855 C6JY7V 11776638 Ki = 17700 nM T15855 C6ET2R 11817181 IC50 = 95000 nM T15855 C19HAP 11825584 IC50 = 126000 nM T15855 CQ0O5A 11952574 IC50 = 43000 nM T15855 CQIB43 11957945 IC50 = 83000 nM T15855 CJAE28 15036410 IC50 = 19000 nM T15855 C6BHJ9 15101668 IC50 > 500000 nM T15855 C2ZMH8 15948988 IC50 = 4756 nM T15855 C13JIX 15949418 IC50 = 5000 nM T15855 C49NUJ 15949507 IC50 = 45600 nM T15855 CU4P5X 15950383 Ki = 886 nM T15855 C16XRI 15950384 Ki > 30000 nM T15855 CUMR27 15950385 Ki = 688 nM T15855 C69RAY 15950386 Ki = 3820 nM T15855 CM63YP 15950387 Ki = 4254 nM T15855 CH8F7W 15950388 Ki = 675 nM T15855 C0L4SH 15950456 Ki > 30000 nM T15855 C8G7OJ 15950457 Ki = 1244 nM T15855 C8FU1V 15950462 Ki > 30000 nM T15855 C9KJ6D 15950538 Ki = 2282 nM T15855 C3C6PM 15950539 Ki = 1039 nM T15855 C4S7AB 15950540 Ki = 3921 nM T15855 C2HGJ0 15950541 Ki = 1708 nM T15855 C3U1VO 15950542 Ki > 30000 nM T15855 CKX8M6 15950615 Ki = 15960 nM T15855 CC0M2X 15951427 Ki = 4504 nM T15855 CF3PX0 15951428 Ki = 3164 nM T15855 CWTX01 15951429 Ki = 1084 nM T15855 C3LQD9 15951431 Ki = 1174 nM T15855 CI3DB4 15951636 IC50 = 1200 nM T15855 CL1E6O 15953860 IC50 > 100000 nM T15855 CLG2Q1 16035093 IC50 > 100000 nM T15855 CMUG74 16035094 IC50 > 100000 nM T15855 C13-MAR 16040457 IC50 > 100000 nM T15855 C0YQ9A 16046127 IC50 = 148000 nM T15855 CS7DQ3 16090844 Ki > 30000 nM T15855 C8CVG9 16090856 Ki > 30000 nM T15855 CU3GB5 16126742 IC50 = 378.8 nM T15855 CHUX72 16202788 Ki > 3000 nM T15855 CC20IT 16203037 Ki > 3000 nM T15855 CA1PV5 16216352 IC50 > 20000 nM T15855 CD9MQ6 16223559 IC50 > 20000 nM T15855 CQ7G8T 16223560 IC50 = 2727 nM T15855 CN24YP 16223762 IC50 > 20000 nM T15855 CF37TH 16226604 IC50 > 20000 nM T15855 C6ANU2 16226605 IC50 > 20000 nM T15855 CFW43X 16658022 IC50 > 100000 nM T15855 C6H5VO 16658023 IC50 > 50000 nM T15855 CC9W4S 16658024 IC50 > 100000 nM T15855 CR51WX 16658101 IC50 > 100000 nM T15855 CMLR19 16658102 IC50 > 100000 nM T15855 CXN32U 16658103 IC50 > 50000 nM T15855 C2XP7B 16658104 IC50 > 100000 nM T15855 CD6L7Z 16658105 IC50 > 100000 nM T15855 C53XZP 16721117 Ki > 3000 nM T15855 CT01PQ 16739331 IC50 = 89120 nM T15855 C61RFP 16755651 IC50 = 3440 nM T15855 CU05RG 17748274 IC50 = 25000 nM T15855 C15TBF 17751406 IC50 = 24 nM T15855 C5W3VY 17753031 IC50 = 49000 nM T15855 CT42AI 20706081 IC50 = 11500 nM T15855 CBZ1E6 21045424 IC50 > 100000 nM T15855 C6ZMS8 21054400 Ki > 3000 nM T15855 CED47V 22690988 IC50 = 23000 nM T15855 C9VGC8 22691359 IC50 > 100000 nM T15855 C1M2ZS 22691666 IC50 > 100000 nM T15855 C8JSI4 23628284 IC50 = 100000 nM T15855 CA95UP 23634434 IC50 > 30000 nM T15855 CAQ81M 23644660 IC50 = 38000 nM T15855 CDPU25 23644665 IC50 > 100000 nM T15855 CCSU21 23645371 IC50 = 210 nM T15855 CFV07G 23645410 IC50 = 45000 nM T15855 CIMG82 23645411 IC50 = 72000 nM T15855 C2Q5IK 23645581 IC50 = 993 nM T15855 C3VA0M 23645582 IC50 > 100000 nM T15855 C1JAG6 23645622 IC50 > 100000 nM T15855 C4B9FM 23645685 Ki = 4 nM T15855 CP9GS5 23645686 IC50 > 100000 nM T15855 C6R2LP 23645687 IC50 > 100000 nM T15855 CN7FK3 23645688 IC50 > 100000 nM T15855 CSHX17 23645689 IC50 > 100000 nM T15855 CL8QV6 23645690 IC50 > 100000 nM T15855 C0AU9X 23645691 IC50 > 100000 nM T15855 CRM3Y4 23645692 IC50 > 100000 nM T15855 CDM8A2 23645693 IC50 > 100000 nM T15855 CIR1F6 23645694 IC50 > 100000 nM T15855 CK5G6I 23645695 IC50 > 100000 nM T15855 CHS76O 23645696 IC50 > 100000 nM T15855 CVP59D 23645697 IC50 > 100000 nM T15855 CH13BW 23645698 IC50 > 100000 nM T15855 CL0K1T 23645699 IC50 > 100000 nM T15855 CB3Z7O 23645700 IC50 > 100000 nM T15855 CNO6Q1 23645702 IC50 > 100000 nM T15855 CGMC54 23645703 IC50 > 100000 nM T15855 C0V4WR 23645705 IC50 > 100000 nM T15855 CY9XW5 23645721 IC50 > 100000 nM T15855 CKM6Y8 23645917 IC50 = 24000 nM T15855 C9Y2ZL 23645918 IC50 = 21000 nM T15855 C4V6BX 23645919 IC50 = 68000 nM T15855 C78PNU 23645920 IC50 > 100000 nM T15855 C5YT6S 23645921 IC50 = 71000 nM T15855 CELQ89 23645922 IC50 > 100000 nM T15855 CGV92H 23645923 IC50 = 18000 nM T15855 CJ60EH 23645924 IC50 = 9400 nM T15855 CZG70A 23645925 IC50 = 72000 nM T15855 CD6V7X 23645926 IC50 = 56000 nM T15855 C1TD4J 23645927 IC50 > 100000 nM T15855 C71PQU 23645928 IC50 = 22000 nM T15855 C8EOB9 23645929 IC50 = 62000 nM T15855 C0M1TH 23645930 IC50 = 58000 nM T15855 CFHB36 23645931 IC50 > 100000 nM T15855 CTG27F 23645932 IC50 = 10000 nM T15855 CS2FT5 23645933 IC50 = 32000 nM T15855 C98QGK 23645934 IC50 = 11000 nM T15855 CS76DY 23645935 IC50 = 65000 nM T15855 C91MYK 23645936 IC50 = 5800 nM T15855 C3AQC0 23645937 IC50 > 100000 nM T15855 C61GTC 23645938 IC50 = 7100 nM T15855 C8XF6R 23645939 IC50 = 29000 nM T15855 C7IX5B 23645940 IC50 = 4300 nM T15855 CP6M3W 23645941 IC50 = 3000 nM T15855 CQ75XK 23645942 IC50 = 3300 nM T15855 C8T7GY 23645943 IC50 = 3200 nM T15855 C25ZXC 23645944 IC50 = 28000 nM T15855 C4A3NI 23645945 IC50 = 51000 nM T15855 C9Y1BP 23646016 IC50 > 20000 nM T15855 CL8DY2 23646017 IC50 > 20000 nM T15855 CT6Q1R 23646018 IC50 > 20000 nM T15855 C8VS1X 23646019 IC50 = 12210 nM T15855 CL4BX5 23646020 IC50 > 20000 nM T15855 CZ24WC 23646021 IC50 > 20000 nM T15855 C98VYW 23646022 IC50 > 20000 nM T15855 CCL17M 23646023 IC50 > 20000 nM T15855 CT16HE 23646024 IC50 > 20000 nM T15855 CAL8T5 23646025 IC50 = 120 nM T15855 CVSH12 23646026 IC50 = 16 nM T15855 C15HJB 23646027 IC50 = 3016 nM T15855 CBUM54 23646029 IC50 > 100000 nM T15855 C32ZNH 23646030 IC50 = 1148 nM T15855 CE8L2I 23646031 IC50 = 78 nM T15855 C8SIU2 23646032 IC50 = 555 nM T15855 C7L6JR 23646033 IC50 = 150 nM T15855 CZ28UC 23646142 Ki > 30000 nM T15855 CLA15H 23646143 Ki = 110 nM T15855 CUZ0D8 23646448 IC50 = 42000 nM T15855 C7PE0S 23646449 IC50 = 13000 nM T15855 COT87G 23646450 IC50 = 21000 nM T15855 CF2J9Q 23646451 IC50 = 53000 nM T15855 C4EG5D 23646512 Ki > 3000 nM T15855 CDM3J0 23646514 Ki > 30000 nM T15855 C5GQ7J 23646519 Ki > 3000 nM T15855 CFOA63 23647106 IC50 = 3000 nM T15855 CFTW63 23647114 IC50 = 38000 nM T15855 C0BQ2D 23647115 IC50 = 29000 nM T15855 CLO1Y2 23647116 IC50 > 100000 nM T15855 CSJ78F 23647117 IC50 = 45000 nM T15855 CDE9L7 23647118 IC50 = 58000 nM T15855 CZF25M 23647119 IC50 = 53000 nM T15855 CW5U3C 23647120 IC50 = 15000 nM T15855 CWO62C 23647121 IC50 = 42000 nM T15855 C0X1CK 23647122 IC50 = 58000 nM T15855 C7JOV9 23647123 IC50 = 93000 nM T15855 C0UT7J 23647124 IC50 = 70000 nM T15855 C8P2VJ 23647125 IC50 = 41000 nM T15855 CQ85KB 23647126 IC50 > 100000 nM T15855 CRFL12 23647127 IC50 = 16000 nM T15855 CP3CF0 23647128 IC50 = 89000 nM T15855 CJA3M7 23647129 IC50 = 26000 nM T15855 C7L3RX 23647130 IC50 = 34000 nM T15855 C8UWB7 23647132 IC50 = 20000 nM T15855 C60MWC 23647133 IC50 = 19000 nM T15855 CBA8N1 23647136 IC50 > 100000 nM T15855 CTB09J 23647311 IC50 > 100000 nM T15855 CJ6XT7 23647314 IC50 > 50000 nM T15855 CO9GD8 23655077 IC50 = 1150 nM T15855 CWVR37 23655298 IC50 = 2110 nM T15855 CPCX60 23655474 IC50 = 16000 nM T15855 CB1E5P 23655476 IC50 = 530 nM T15855 CWTD09 23655478 IC50 = 48000 nM T15855 CW9UR3 23657402 IC50 = 36000 nM T15855 CU18EA 23657547 IC50 = 17500 nM T15855 CVF6E2 23661697 IC50 > 100000 nM T15855 CM7C4W 23661708 IC50 = 30000 nM T15855 CO6L9F 23661716 IC50 > 100000 nM T15855 CHR14F 23661718 IC50 > 100000 nM T15855 CNP9T1 24180585 IC50 = 3200 nM T15855 CI0W8A 24755210 IC50 = 460000 nM T15855 CX8DH1 24769723 IC50 > 100000 nM T15855 C0H8OB 24776705 IC50 > 100000 nM T15855 C24GLZ 24776939 IC50 = 332 nM T15855 C6LD2J 24777439 IC50 > 100000 nM T15855 CK8EL5 24777568 IC50 = 70000 nM T15855 CQ20PV 24777692 IC50 > 100000 nM T15855 C1WF3I 24777804 IC50 = 17000 nM T15855 C50SPA 24784161 IC50 = 71 nM T15855 C29SZR 24784416 IC50 = 120 nM T15855 C0H8IZ 24784426 IC50 = 177 nM T15855 CO7L6R 24784427 IC50 = 2196 nM T15855 C8FQT4 24784664 IC50 = 5962 nM T15855 C69QMZ 24784674 IC50 = 389 nM T15855 CW8LK2 24784675 IC50 = 439 nM T15855 CH1W5N 24784676 IC50 = 1412 nM T15855 CJ0ZI7 24784677 IC50 = 13217 nM T15855 CIZF59 24784915 IC50 = 1439 nM T15855 CKFH56 24784916 IC50 = 2712 nM T15855 C5HY0P 24784918 IC50 = 3055 nM T15855 CS6HU2 24784925 IC50 = 2110 nM T15855 CK6W8S 24784926 IC50 = 174 nM T15855 CUH32V 24785152 IC50 = 1597 nM T15855 C2KL7G 24794725 IC50 = 19 nM T15855 CUM03S 24798754 IC50 = 44000 nM T15855 CZ3ND1 24832041 IC50 > 100000 nM T15855 CY9W8O 24860300 IC50 = 21000 nM T15855 CMK9B7 24894026 IC50 = 160 nM T15855 CYL69J 24951732 IC50 = 91000 nM T15855 CNP3T1 24951733 IC50 = 8600 nM T15855 CDCP18 24952087 IC50 = 79000 nM T15855 CIM7S2 24952089 IC50 = 100000 nM T15855 CX83WL 24963343 IC50 > 100000 nM T15855 CA94RD 24999327 IC50 = 17380 nM T15855 CZJ2N6 24999330 IC50 = 18240 nM T15855 C01GPL 25132159 Ki = 880 nM T15855 C7IDX9 25132160 Ki = 96 nM T15855 C9VK8W 25132161 Ki = 140 nM T15855 CFZ4V2 25132162 Ki = 8400 nM T15855 CSU0B5 25189891 IC50 > 30000 nM T15855 C7KN2U 42608447 IC50 = 5700 nM T15855 C60SVD 42636924 IC50 > 20000 nM T15855 CS40ML 44123747 IC50 > 50000 nM T15855 CQF86D 44182505 IC50 = 4890 nM T15855 C3I4TF 44201003 IC50 > 100000 nM T15855 CE5B7H 44218404 IC50 > 20000 nM T15855 CR8GT4 44218550 IC50 > 20000 nM T15855 CBW7D4 44218551 IC50 > 20000 nM T15855 CVH08B 44218552 IC50 > 20000 nM T15855 CISE95 44218553 IC50 > 20000 nM T15855 CLB72R 44218554 IC50 > 20000 nM T15855 C2N9VR 44218555 IC50 > 20000 nM T15855 CJ6L3S 44218693 IC50 > 20000 nM T15855 C97IFE 44218695 IC50 > 20000 nM T15855 C50EKW 44250174 IC50 = 5200 nM T15855 CRZI12 44266022 IC50 = 530 nM T15855 CFY7P3 44360924 IC50 = 170 nM T15855 CA7KI2 44390794 IC50 > 100000 nM T15855 CW81MP 44394103 IC50 = 2100 nM T15855 C1VLP6 44399148 IC50 = 2327 nM T15855 CIED90 44399244 IC50 = 28 nM T15855 C3PKV8 44399546 IC50 = 220 nM T15855 CPX1M9 44403336 IC50 = 1000 nM T15855 CSEN70 44403337 IC50 = 190 nM T15855 C91MNA 44403353 IC50 = 4300 nM T15855 CR53EK 44403354 IC50 = 2600 nM T15855 C8MLN6 44403355 IC50 = 350 nM T15855 CRO16Q 44403360 IC50 = 30 nM T15855 C0FC7D 44403361 IC50 = 95 nM T15855 C41IAB 44403437 IC50 = 6000 nM T15855 CCOA39 44403438 IC50 = 400 nM T15855 CLYJ80 44403439 IC50 = 5200 nM T15855 CGJ17L 44415883 IC50 = 65000 nM T15855 CE0KW2 44415905 IC50 > 100000 nM T15855 CPR49A 44415906 IC50 > 100000 nM T15855 CQ5P2J 44415929 IC50 > 100000 nM T15855 CM2W5X 44415930 IC50 > 100000 nM T15855 COPZ87 44415944 IC50 > 500000 nM T15855 CSG4F8 44417393 Ki = 5200 nM T15855 CE7UB0 44418114 IC50 = 80000 nM T15855 C70KAO 44418211 IC50 = 1473 nM T15855 C8LC2A 44418213 IC50 > 20000 nM T15855 CTM1Y8 44418214 IC50 > 20000 nM T15855 C1EMA5 44418215 IC50 > 20000 nM T15855 CWDH12 44418216 IC50 > 20000 nM T15855 C1FB4K 44418218 IC50 > 20000 nM T15855 CVC3R4 44418219 IC50 > 20000 nM T15855 CU1FG2 44418222 IC50 > 20000 nM T15855 C8ZH5R 44418223 IC50 > 20000 nM T15855 CA9YM3 44418225 IC50 > 20000 nM T15855 CQE5Y0 44418229 IC50 > 20000 nM T15855 C2LXS7 44418232 IC50 > 20000 nM T15855 C59HZQ 44418251 IC50 = 11000 nM T15855 C2UR9X 44418256 IC50 > 20000 nM T15855 CK20CA 44418257 IC50 > 20000 nM T15855 CO3GL6 44418260 IC50 > 20000 nM T15855 CY3O7C 44418261 IC50 > 20000 nM T15855 C0ITV9 44418262 IC50 > 20000 nM T15855 C68SHD 44418264 IC50 > 20000 nM T15855 CDI98V 44418265 IC50 > 20000 nM T15855 CHO5P1 44418266 IC50 > 20000 nM T15855 C95XQC 44418268 IC50 > 20000 nM T15855 C0FT8Q 44420999 Ki > 30000 nM T15855 C6NV0S 44421004 Ki = 19100 nM T15855 C5W8VX 44421005 Ki > 30000 nM T15855 C9IRG5 44422418 IC50 = 736.5 nM T15855 CS63GZ 44422443 IC50 = 562.8 nM T15855 CNQC83 44422485 IC50 = 678.9 nM T15855 CZ2MB8 44426068 IC50 = 46000 nM T15855 C8PKO5 44426070 IC50 = 76000 nM T15855 C7IL3S 44431164 IC50 = 75000 nM T15855 C0UOS8 44431165 IC50 > 100000 nM T15855 CEG05S 44431166 IC50 = 65000 nM T15855 CO8S3Z 44431170 IC50 > 10000 nM T15855 C2K4RQ 44431176 IC50 > 10000 nM T15855 CJZY21 44431177 IC50 > 10000 nM T15855 CSJI40 44431185 IC50 > 100000 nM T15855 C36EJR 44431188 IC50 > 100000 nM T15855 C2MCA1 44431191 IC50 > 100000 nM T15855 C89XVB 44431197 IC50 > 100000 nM T15855 CK76EP 44431199 IC50 > 100000 nM T15855 C3FPT2 44431200 IC50 > 100000 nM T15855 C4F8AG 44431201 IC50 = 26000 nM T15855 CWX4I3 44431203 IC50 > 100000 nM T15855 CZ3N9E 44431204 IC50 = 30000 nM T15855 C5NAS6 44431205 IC50 > 100000 nM T15855 C37SGU 44431206 IC50 > 100000 nM T15855 CYD62G 44431212 IC50 = 979 nM T15855 C72WTP 44431213 IC50 = 1010 nM T15855 CC3T9G 44431214 IC50 = 4200 nM T15855 CL4T3X 44431215 IC50 = 37000 nM T15855 C4WVL8 44431216 IC50 > 100000 nM T15855 CO08HZ 44431217 IC50 = 39000 nM T15855 CCPZ23 44431218 IC50 = 54000 nM T15855 C0J7WV 44431219 IC50 = 86000 nM T15855 C16ZTV 44431220 IC50 > 22000 nM T15855 CR0A1M 44431316 IC50 > 100000 nM T15855 CV1R7A 44431317 IC50 > 100000 nM T15855 CY76AB 44432858 IC50 = 67300 nM T15855 CS95EU 44432859 IC50 = 69900 nM T15855 C1PX9V 44432860 IC50 = 6590 nM T15855 CE4Q5X 44432862 IC50 = 1450 nM T15855 CHN6E3 44432863 IC50 = 5720 nM T15855 CF2AT6 44432881 IC50 < 390 nM T15855 CTD24F 44432889 IC50 < 390 nM T15855 CU67PL 44432901 IC50 = 5800 nM T15855 C35GZP 44432904 IC50 = 808 nM T15855 C21UQD 44432911 IC50 = 1440 nM T15855 CU27DF 44432914 IC50 = 3260 nM T15855 C9E1SZ 44432915 IC50 = 4400 nM T15855 CZ47KB 44432929 IC50 < 390 nM T15855 CS5BT9 44432935 IC50 = 1290 nM T15855 CI9M8R 44432936 IC50 < 390 nM T15855 C5LTR0 44432937 IC50 < 390 nM T15855 C6EJB0 44432938 IC50 < 390 nM T15855 CJ7YN0 44432940 IC50 = 3100 nM T15855 CVZ3I2 44432942 IC50 = 930 nM T15855 CT29BC 44432944 IC50 = 1090 nM T15855 CQDS95 44433224 IC50 = 1600 nM T15855 C9GIE3 44433617 IC50 = 25000 nM T15855 C5B4HS 44433618 IC50 = 3600 nM T15855 CU6XZ5 44433646 IC50 > 100000 nM T15855 CM8E2D 44433661 IC50 = 22000 nM T15855 CE92DA 44435310 IC50 = 86000 nM T15855 C3SBK5 44435313 IC50 = 910 nM T15855 CX7UN0 44435314 IC50 = 43000 nM T15855 CE7XI5 44435315 IC50 = 7800 nM T15855 CGAR49 44435316 IC50 = 12500 nM T15855 CEL4H9 44439337 IC50 = 12 nM T15855 C0OJ1T 44439353 IC50 = 40 nM T15855 C08ZST 44440659 Ki > 3000 nM T15855 CR3PM7 44440662 Ki = 4320 nM T15855 CB4Q0H 44440663 Ki = 6440 nM T15855 CCSI57 44440665 Ki = 4350 nM T15855 CR4B1M 44443293 IC50 = 27400 nM T15855 CY16JP 44443294 IC50 = 26400 nM T15855 CN24IJ 44443296 IC50 > 30000 nM T15855 C8DSC1 44443297 IC50 = 23100 nM T15855 C4F5JW 44443298 IC50 > 30000 nM T15855 CJ0G3N 44443299 IC50 > 30000 nM T15855 C9F7NQ 44443300 IC50 = 10200 nM T15855 C7QCO2 44443301 IC50 = 24100 nM T15855 CCQ82F 44443302 IC50 = 4250 nM T15855 C1M5TF 44443309 IC50 = 5100 nM T15855 CSAE59 44443313 IC50 = 1200 nM T15855 CK5E8V 44443319 IC50 = 4700 nM T15855 CD0NM4 44443335 IC50 = 3100 nM T15855 CEF6H5 44443336 IC50 = 2500 nM T15855 CTIM25 44443338 IC50 = 1900 nM T15855 CE9Q7A 44443341 IC50 = 1800 nM T15855 CI8Q5O 44443343 IC50 = 1000 nM T15855 C0MOV3 44443346 IC50 = 560000 nM T15855 C52VPZ 44443347 IC50 = 461000 nM T15855 CJ8P7U 44443348 IC50 = 148000 nM T15855 C8U1XN 44443349 IC50 = 922000 nM T15855 CM5WU9 44443350 IC50 = 858000 nM T15855 CB9IM0 44443351 IC50 = 247000 nM T15855 C8WI4F 44443352 IC50 = 3290000 nM T15855 C3NI8P 44443353 IC50 = 326000 nM T15855 C7M0HV 44443354 IC50 = 704000 nM T15855 C0UG4R 44443355 IC50 = 363000 nM T15855 C7B5HK 44443356 IC50 = 190000 nM T15855 C2G1PX 44443357 IC50 = 586000 nM T15855 C3AUF2 44443358 IC50 = 258000 nM T15855 C0WO5B 44443359 IC50 = 1150000 nM T15855 CUG6X5 44443360 IC50 = 1040000 nM T15855 CARK80 44443361 IC50 = 332000 nM T15855 CP7WL5 44443363 IC50 = 346000 nM T15855 C4V0SN 44443364 IC50 = 417000 nM T15855 CD2L9G 44443366 IC50 = 203000 nM T15855 CA0NZ7 44443707 IC50 = 9400 nM T15855 C24ZHB 44443708 IC50 = 68000 nM T15855 C8R4OD 44443709 IC50 = 50000 nM T15855 CLDN63 44443710 IC50 = 58000 nM T15855 C7LNP2 44443711 IC50 = 77000 nM T15855 CJX2M7 44443712 IC50 = 54000 nM T15855 C6RST0 44443713 IC50 > 100000 nM T15855 C3YL9X 44443714 IC50 = 23000 nM T15855 CRH8M1 44443715 IC50 > 100000 nM T15855 CIB50E 44443717 IC50 = 6600 nM T15855 CK6QF4 44443719 IC50 = 26000 nM T15855 CX6O1P 44443720 IC50 = 64000 nM T15855 C0YV2D 44443723 IC50 = 55000 nM T15855 C1BUJ5 44443725 IC50 = 4000 nM T15855 CXS34I 44443727 IC50 = 39000 nM T15855 CCHS17 44443729 IC50 = 85000 nM T15855 C39KZG 44443736 IC50 = 33000 nM T15855 C5H8EJ 44443737 IC50 = 80000 nM T15855 CS3Y1G 44444344 IC50 > 100000 nM T15855 CL2U9C 44444352 IC50 = 44000 nM T15855 C8VE5T 44444353 IC50 > 100000 nM T15855 C8F5HC 44444371 IC50 = 25000 nM T15855 CEW50M 44444373 IC50 = 16000 nM T15855 CO0M7Y 44444375 IC50 = 71000 nM T15855 CS93BI 44444377 IC50 = 86000 nM T15855 C9J4FB 44444379 IC50 > 100000 nM T15855 C3YA4K 44444383 IC50 > 100000 nM T15855 C75OIP 44444386 IC50 > 100000 nM T15855 C4J6ZG 44444390 IC50 > 100000 nM T15855 C05EBU 44444391 IC50 > 100000 nM T15855 CSN27E 44445042 IC50 = 1600 nM T15855 CGN61Q 44445047 IC50 = 3000 nM T15855 CYW8E3 44445051 IC50 = 30000 nM T15855 CRG64M 44445053 IC50 = 622 nM T15855 C6ZID3 44445055 IC50 = 367 nM T15855 C72KOR 44445057 IC50 = 8000 nM T15855 C0RTA6 44445060 IC50 = 1103 nM T15855 CIK8G3 44445063 IC50 = 326 nM T15855 CN05VX 44445065 IC50 > 100000 nM T15855 COA90R 44445067 IC50 = 5000 nM T15855 C91DWY 44560396 IC50 = 7300 nM T15855 CZ9WJ0 44560397 IC50 > 100000 nM T15855 C0FLU7 44560398 IC50 = 1200 nM T15855 CX9BK6 44560399 IC50 = 202 nM T15855 CZ43JR 44560454 IC50 = 4600 nM T15855 CY38QP 44560549 IC50 > 100000 nM T15855 C7IL3K 44560550 IC50 > 100000 nM T15855 CF9J7Z 44560551 IC50 = 4900 nM T15855 C1QAI4 44560552 IC50 > 25000 nM T15855 CK25CG 44560553 IC50 > 50000 nM T15855 C4C9NG 44560554 IC50 > 100000 nM T15855 CKIH45 44560555 IC50 = 56900 nM T15855 C2LW3C 44560595 IC50 = 800 nM T15855 C47WCK 44560596 IC50 = 2800 nM T15855 CL8AE5 44560597 IC50 > 100000 nM T15855 C1YJ8C 44560648 IC50 = 111 nM T15855 CY6GU1 44560649 IC50 = 666 nM T15855 C12EYZ 44560650 IC50 = 43 nM T15855 C7LY9V 44560651 IC50 = 479 nM T15855 CG5CB2 44560698 IC50 = 2900 nM T15855 CR56BA 44560699 IC50 = 710 nM T15855 CIA45R 44560700 IC50 = 12000 nM T15855 CAK3U5 44560701 IC50 = 910 nM T15855 CJE42H 44560746 IC50 = 10200 nM T15855 C5OW2C 44560747 IC50 = 24000 nM T15855 CM2GN5 44560748 IC50 = 5900 nM T15855 C5FSB4 44560749 IC50 = 13000 nM T15855 C5WEG1 44560750 IC50 = 290 nM T15855 CN0KO4 44560770 IC50 = 51 nM T15855 CZSO82 44560823 IC50 = 41000 nM T15855 C4IVD9 44560824 IC50 = 6800 nM T15855 C4L3VZ 44560825 IC50 = 1100 nM T15855 CHV7S1 44560826 IC50 = 5700 nM T15855 CE3NF4 44560849 IC50 = 1900 nM T15855 CT6P5E 44560850 IC50 = 12000 nM T15855 CTH9P2 44560851 IC50 = 5600 nM T15855 CGZ48C 44560928 IC50 = 5200 nM T15855 C9EK8A 44560929 IC50 = 312000 nM T15855 CM68VD 44560930 IC50 = 520 nM T15855 C4SMJ1 44560961 IC50 = 240 nM T15855 C2I3TR 44560962 IC50 = 72 nM T15855 CGV49L 44560963 IC50 = 11 nM T15855 CY0L1G 44560964 IC50 = 71 nM T15855 C7FST1 44560988 IC50 = 21 nM T15855 CGOM86 44560989 IC50 = 22000 nM T15855 C74ZNK 44560990 IC50 = 187 nM T15855 C95AUS 44560991 IC50 = 13.8 nM T15855 CTJ23N 44561008 IC50 > 100000 nM T15855 CR2A0E 44561009 IC50 = 64000 nM T15855 C4LQY2 44561010 IC50 > 100000 nM T15855 C28XDF 44561011 IC50 > 100000 nM T15855 CQ04BE 44561046 IC50 = 17000 nM T15855 C8IF7B 44561117 IC50 = 18000 nM T15855 C29VDX 44561118 IC50 = 27000 nM T15855 CB4JA7 44561119 IC50 = 47000 nM T15855 C5K9CX 44561120 IC50 > 100000 nM T15855 CQ8DN4 44561152 IC50 > 100000 nM T15855 C4DBU1 44561153 IC50 > 100000 nM T15855 C73WBR 44561154 IC50 > 100000 nM T15855 CJ91UC 44561155 IC50 > 100000 nM T15855 CMO6S2 44561191 IC50 = 41000 nM T15855 CF9SB3 44561192 IC50 = 87000 nM T15855 C5X1VJ 44561193 IC50 = 15000 nM T15855 C31GMV 44561194 IC50 = 27000 nM T15855 C1U4YQ 44565237 IC50 = 11000 nM T15855 CRK69O 44565238 IC50 > 20000 nM T15855 C6M2WD 44565239 IC50 = 8600 nM T15855 CTZ9L0 44565254 IC50 > 20000 nM T15855 CEMV93 44565274 IC50 > 20000 nM T15855 C5E6PQ 44565275 IC50 > 20000 nM T15855 CI93OK 44565276 IC50 > 20000 nM T15855 C2HRF1 44565277 IC50 = 12000 nM T15855 CFEC28 44565466 IC50 > 20000 nM T15855 C5MON6 44565467 IC50 > 20000 nM T15855 CGA4U6 44565488 IC50 > 20000 nM T15855 C1BZ3I 44565489 IC50 > 20000 nM T15855 CP3C5F 44565490 IC50 > 20000 nM T15855 CRU86T 44565491 IC50 > 20000 nM T15855 C3C2DL 44565492 IC50 > 20000 nM T15855 CJ2W1P 44565512 IC50 > 20000 nM T15855 C5Z9GW 44565513 IC50 > 20000 nM T15855 C3I0MO 44565514 IC50 > 20000 nM T15855 CI3J6Y 44565535 IC50 > 20000 nM T15855 CB90XZ 44565536 IC50 > 20000 nM T15855 C01SLH 44565537 IC50 > 20000 nM T15855 C8Y2LX 44565538 IC50 > 20000 nM T15855 CXD19F 44565539 IC50 > 20000 nM T15855 CFK92H 44565583 IC50 = 7880 nM T15855 CA0O7F 44565585 IC50 > 30000 nM T15855 CPZ7J3 44565844 IC50 = 2240 nM T15855 C9BGR3 44565845 IC50 = 2660 nM T15855 CR83QA 44565869 IC50 = 970 nM T15855 C6K2WL 44565870 IC50 = 540 nM T15855 C3UL2E 44565871 IC50 = 530 nM T15855 C9SL5D 44565872 IC50 = 9150 nM T15855 CZBX95 44565889 IC50 = 9690 nM T15855 C1TLY0 44565890 IC50 = 10300 nM T15855 CEO20N 44565891 IC50 = 15100 nM T15855 COA7X5 44565892 IC50 = 17100 nM T15855 CRO3D2 44567651 IC50 = 14900 nM T15855 CM95OD 44567652 IC50 = 13100 nM T15855 CX6WL5 44567653 IC50 = 837 nM T15855 C4MP9D 44567654 IC50 = 2375 nM T15855 CV23FP 44567668 IC50 = 1667 nM T15855 CD4C7Y 44567710 IC50 = 35500 nM T15855 C4CUJ6 44567711 IC50 = 2180 nM T15855 CK1C7W 44567712 IC50 = 3400 nM T15855 CTK1I9 44567713 IC50 = 16100 nM T15855 CM50CU 44567747 IC50 = 10100 nM T15855 CNA0I9 44567918 IC50 = 2210 nM T15855 C6BXT0 44567919 IC50 = 637 nM T15855 CJ85MG 44567920 IC50 = 3030 nM T15855 CUJD19 44567976 IC50 = 1675 nM T15855 C5YB6E 44567977 IC50 = 399 nM T15855 CNF09E 44567978 IC50 = 3020 nM T15855 C70WEI 44567979 IC50 = 652 nM T15855 CW7NB6 44568016 IC50 = 500 nM T15855 CY8Z3F 44568017 IC50 = 2080 nM T15855 CRM76D 44568018 IC50 = 2130 nM T15855 CCG83U 44568057 IC50 = 2400 nM T15855 C8XW9A 44568058 IC50 > 10000 nM T15855 CMQ7D5 44568097 IC50 = 6500 nM T15855 C1F9OL 44568098 IC50 = 366 nM T15855 CUYK75 44568099 IC50 > 10000 nM T15855 CZ81XF 44568100 IC50 = 28600 nM T15855 C6GT0A 44568134 IC50 = 3090 nM T15855 C6IW5D 44568135 IC50 = 2050 nM T15855 C3PWD8 44568136 IC50 = 3270 nM T15855 C4NCA7 44568169 IC50 = 4030 nM T15855 C8TXH9 44568170 IC50 = 11100 nM T15855 C17PZX 44568171 IC50 = 11499 nM T15855 C7SCJ1 44568172 IC50 = 7270 nM T15855 CZCU54 44571949 IC50 = 4265 nM T15855 CJ96CO 44571951 IC50 = 18197 nM T15855 C7E6IB 44572718 IC50 = 220 nM T15855 CUH81Y 44572719 IC50 = 1200 nM T15855 CJHR19 44572720 IC50 = 360 nM T15855 CG71OU 44572782 IC50 > 20000 nM T15855 C2DQ0C 44589933 IC50 = 49000 nM T15855 CUZ3P0 44589935 IC50 = 45800 nM T15855 CBAH06 44590649 IC50 = 1700 nM T15855 CRN4U5 44590696 IC50 > 100000 nM T15855 CY8R3Q 44593399 IC50 = 1320 nM T15855 CP8YC3 44593408 IC50 = 200 nM T15855 C4L6NS 44593409 IC50 = 200 nM T15855 CI0FT1 44593463 IC50 > 20000 nM T15855 C65KPR 45101722 IC50 = 18300 nM T15855 CXYT36 45101723 IC50 = 10000 nM T15855 C2RNP7 45102670 IC50 = 41000 nM T15855 CGZD98 45265711 IC50 = 35000 nM T15855 CW09DZ 45265891 Ki > 3000 nM T15855 CCO76A 45266134 IC50 = 63000 nM T15855 CU4C5P 45266135 IC50 > 100000 nM T15855 CLVM20 45266136 IC50 = 12000 nM T15855 C8H9GV 45267527 IC50 = 2300 nM T15855 CP9B0W 45267530 IC50 = 1200 nM T15855 C3GJK0 45267531 IC50 = 3000 nM T15855 CN38QU 45268229 IC50 = 4000 nM T15855 CEQ16V 45268233 IC50 = 200 nM T15855 C0QB1V 45268417 IC50 = 3100 nM T15855 C2S9ZT 45268436 IC50 = 6400 nM T15855 CX8WC0 45269123 IC50 = 4200 nM T15855 C9HR0K 45269274 IC50 = 8200 nM T15855 CZ1N2O 45269275 IC50 = 7300 nM T15855 CIE21V 45269276 IC50 = 6000 nM T15855 CWT60M 45269971 IC50 = 22000 nM T15855 C8QJ7X 45270108 IC50 = 3900 nM T15855 CYWK62 45270115 IC50 = 7900 nM T15855 CGF7Z6 45270958 IC50 = 9000 nM T15855 CH5S8Y 45270959 IC50 = 10000 nM T15855 C5NH6Q 45271791 IC50 = 2400 nM T15855 C8Z3DK 45271794 IC50 = 4900 nM T15855 CX62YA 45271796 IC50 = 9900 nM T15855 CZ8EO2 45271803 IC50 = 9200 nM T15855 CJ7Q9E 45271813 IC50 = 6000 nM T15855 CJI2R6 45272664 IC50 = 4200 nM T15855 C49BKQ 45272672 IC50 = 7800 nM T15855 CP36CT 45272682 IC50 = 3500 nM T15855 C8NL4U 45272683 IC50 = 5900 nM T15855 C6S0OC 45273404 IC50 = 7300 nM T15855 CYMR87 45273573 IC50 = 2300 nM T15855 CFL87A 45273581 IC50 = 3000 nM T15855 C2XB0P 45273589 IC50 = 3400 nM T15855 C28PRV 45273594 IC50 = 7000 nM T15855 CSX2T9 45273602 IC50 = 31000 nM T15855 CMP59Q 45273603 IC50 = 6600 nM T15855 C4MFG7 45481845 IC50 = 21000 nM T15855 C28ZXW 45487888 IC50 = 52000 nM T15855 C2N3IZ 45487894 IC50 = 37000 nM T15855 CP62TC 45487898 IC50 = 34000 nM T15855 CWQ1R9 45487903 IC50 = 8200 nM T15855 C8H1KY 45487904 IC50 = 21000 nM T15855 C6X7WJ 45487908 IC50 = 27000 nM T15855 C5OXM9 45487915 IC50 = 23000 nM T15855 CPJ19X 45487917 IC50 = 72000 nM T15855 CV2R7M 45487920 IC50 = 13000 nM T15855 C57JRG 45487921 IC50 = 26000 nM T15855 C4JD1P 45487922 IC50 = 25000 nM T15855 CPB85R 45487926 IC50 = 35000 nM T15855 CTY16E 45487930 IC50 = 26000 nM T15855 C4QTL9 45487931 IC50 = 18000 nM T15855 CG9V0L 45487940 IC50 = 41000 nM T15855 C5XTV1 45487945 IC50 = 2500 nM T15855 C3VK4G 45487946 IC50 = 4500 nM T15855 C0SNL2 46209134 IC50 > 100000 nM T15855 CE9M5C 46209244 IC50 = 60000 nM T15855 CW60IG 46209246 IC50 > 100000 nM T15855 CDP7Q4 46870369 IC50 = 3350 nM T15855 CPH7B4 46871723 IC50 = 23 nM T15855 CDBC45 46890720 IC50 > 20000 nM T15855 CLK47C 46890721 IC50 > 20000 nM T15855 CS6HL3 46890722 IC50 > 20000 nM T15855 C2JY6P 46890723 IC50 > 20000 nM T15855 CP7C1L 46890780 IC50 > 20000 nM T15855 CED80Z 46890852 IC50 > 20000 nM T15855 CA3PE4 46890853 IC50 > 20000 nM T15855 CY9T8W 46890854 IC50 > 20000 nM T15855 C3TJ0H 46890912 IC50 > 20000 nM T15855 CT9HQ6 46890913 IC50 > 20000 nM T15855 C9IP7B 46890914 IC50 > 20000 nM T15855 CSZE87 46891193 IC50 = 7930 nM T15855 C18UES 46891235 IC50 = 3740 nM T15855 C23LCY 46891237 IC50 = 8420 nM T15855 C57UXS 46891239 IC50 = 12740 nM T15855 CJ4G6X 46891342 IC50 = 1430 nM T15855 CAL9K6 46891534 IC50 > 20000 nM T15855 CPN5T2 46891535 IC50 > 20000 nM T15855 C4XTW7 46893990 IC50 > 100000 nM T15855 C8O5VR 46899592 Ki = 13 nM T15855 CTY0M5 46899593 Ki = 2.8 nM T15855 CK9TH1 46899594 Ki = 1.3 nM T15855 C8XD0Q 46899595 Ki = 2 nM T15855 CZ84ST 46899596 Ki = 0.42 nM T15855 CPZ70E 46899597 Ki = 2.2 nM T15855 CD3IJ8 46899752 Ki = 0.7 nM T15855 CRK59N 46899753 Ki = 2.3 nM T15855 C6LXU5 46899754 Ki = 2.9 nM T15855 C52JZL 46899755 Ki = 1.1 nM T15855 C4RC1S 46899756 Ki = 4.1 nM T15855 CP84HR 46899757 Ki = 1.7 nM T15855 CBV4W0 46899937 Ki = 0.4 nM T15855 C5QEJ4 46899938 Ki = 1.3 nM T15855 CHR6V9 46899939 Ki = 4.5 nM T15855 CQ3A8F 46899940 Ki = 2.5 nM T15855 CX2P8Z 46899941 Ki = 0.95 nM T15855 CC2X1J 46899942 Ki = 1.1 nM T15855 C5QA9M 46900103 Ki = 1.4 nM T15855 CBI0Q2 46900104 Ki = 1.2 nM T15855 C4IU2E 46900105 Ki = 0.65 nM T15855 CZEB71 46900106 Ki = 2.2 nM T15855 C2TJW5 46900108 Ki = 0.6 nM T15855 C54ATK 46900259 Ki = 0.58 nM T15855 CI3P6J 46900261 Ki = 1.7 nM T15855 C6DP2G 46900418 Ki = 2.2 nM T15855 CP50DR 46900420 Ki > 10 nM T15855 C8DSG7 46916343 IC50 > 100000 nM T15855 C3RO8F 46916345 IC50 > 100000 nM T15855 CX07LJ 46916346 IC50 > 100000 nM T15855 CF94MW 46916347 IC50 > 100000 nM T15855 CH3F7O 46916384 IC50 > 100000 nM T15855 CM8W6E 46916385 IC50 > 100000 nM T15855 C6FA9Q 46916386 IC50 > 100000 nM T15855 CAW86J 46916387 IC50 > 100000 nM T15855 C63HBE 46916388 IC50 > 100000 nM T15855 CD1CZ7 46916389 IC50 > 100000 nM T15855 CH80LK 46916433 IC50 > 100000 nM T15855 CN4A3P 46916435 IC50 > 100000 nM T15855 CUQ86M 46917047 IC50 > 100000 nM T15855 CS5X9L 46917048 IC50 > 100000 nM T15855 CZP24U 46917049 IC50 = 500 nM T15855 CGMJ52 46938499 IC50 > 100000 nM T15855 C5RAS7 46938602 IC50 > 100000 nM T15855 C3B1LX 46938704 IC50 > 100000 nM T15855 C5TU1F 46938705 IC50 > 100000 nM T15855 CAGP83 46938706 IC50 > 100000 nM T15855 CP9V8Q 46938799 IC50 > 100000 nM T15855 CAB2H9 46938802 IC50 > 100000 nM T15855 CR5X3K 49785099 IC50 > 25000 nM T15855 C2HU0V 49785100 IC50 > 25000 nM T15855 CX7M2K 49785101 IC50 > 25000 nM T15855 C3XCV4 49785102 IC50 > 25000 nM T15855 CZ7A9E 49796933 IC50 > 100000 nM T15855 C5RF0Y 49796938 IC50 = 4100 nM T15855 CE0C3Y 49796939 IC50 > 100000 nM T15855 CI4ZE6 49796940 IC50 > 50000 nM T15855 CBD8K2 49796942 IC50 > 100000 nM T15855 CI25XP 49796945 IC50 = 5300 nM T15855 C8WYA5 49796953 IC50 > 100000 nM T15855 CQH86V 49796955 IC50 > 100000 nM T15855 CBMV50 49796972 IC50 = 87000 nM T15855 C8IL0K 49796973 IC50 > 100000 nM T15855 CA90LB 49796974 IC50 = 16000 nM T15855 C07DHG 49796977 IC50 = 49000 nM T15855 CAS2P4 49796982 IC50 > 100000 nM T15855 CG79KT 49796985 IC50 > 100000 nM T15855 C4D8RE 49796990 IC50 > 100000 nM T15855 CUKB68 49796994 IC50 > 100000 nM T15855 CUR9B0 49796995 IC50 = 15000 nM T15855 CWHO58 49796998 IC50 = 27000 nM T15855 CX74RG 49796999 IC50 > 100000 nM T15855 C20MAQ 49797000 IC50 = 40000 nM T15855 CD67OX 49797001 IC50 > 100000 nM T15855 C9LEF5 49797002 IC50 = 13000 nM T15855 CO2AX9 49797003 IC50 = 2100 nM T15855 CEM61W 49797006 IC50 > 100000 nM T15855 C7Y0JL 49797007 IC50 = 52000 nM T15855 CW45IK 49797008 IC50 = 41000 nM T15855 C79JUI 49797011 IC50 = 22000 nM T15855 CVAK94 49797012 IC50 > 100000 nM T15855 CUK5J1 49797013 IC50 = 460 nM T15855 C4ZK5C 49797014 IC50 > 100000 nM T15855 C1PV8J 49797015 IC50 = 37000 nM T15855 C9YEU6 49797016 IC50 > 100000 nM T15855 CZD4S2 49797017 IC50 = 26000 nM T15855 CKY80F 49797018 IC50 = 19000 nM T15855 CS0D8Q 49797021 IC50 = 8000 nM T15855 C3GF4M 49797022 IC50 > 100000 nM T15855 C8XZT9 49797023 IC50 = 26000 nM T15855 C5H2AS 49797024 IC50 = 32000 nM T15855 C4P0VW 49797025 IC50 = 18000 nM T15855 CVY8M1 49797028 IC50 > 100000 nM T15855 CM59HB 49797029 IC50 > 100000 nM T15855 CH7Y1J 49797030 IC50 = 47000 nM T15855 CX18HI 49797031 IC50 = 14000 nM T15855 CUM28Z 49797035 IC50 > 100000 nM T15855 COS23G 49797036 IC50 = 22000 nM T15855 C2TSG6 49797038 IC50 = 6900 nM T15855 C7BI3W 49797039 IC50 > 100000 nM T15855 C71THK 49797040 IC50 > 100000 nM T15855 C0SG5O 49797041 IC50 > 100000 nM T15855 CM37VB 49797042 IC50 > 100000 nM T15855 C51NUG 49797043 IC50 > 100000 nM T15855 C65WXC 49797044 IC50 > 100000 nM T15855 CHTO37 49797045 IC50 > 100000 nM T15855 CA8R5K 49797046 IC50 > 100000 nM T15855 CLAR35 49797047 IC50 > 100000 nM T15855 C9OCZ3 49797048 IC50 > 100000 nM T15855 C49RUW 49797049 IC50 > 100000 nM T15855 C4EHT7 49797050 IC50 > 100000 nM T15855 CW6G5R 49797051 IC50 = 57000 nM T15855 CUK6G0 49797052 IC50 = 85000 nM T15855 CJ1FE2 49797053 IC50 > 100000 nM T15855 CKJO08 49797054 IC50 > 100000 nM T15855 C70KVU 49797055 IC50 > 100000 nM T15855 CP59BI 49797056 IC50 = 61000 nM T15855 CEDL61 49797057 IC50 > 100000 nM T15855 C5J2LV 49797058 IC50 > 100000 nM T15855 CEI20Q 49797059 IC50 > 100000 nM T15855 C7B5DY 49797060 IC50 > 100000 nM T15855 C5B1RM 49797061 IC50 > 100000 nM T15855 C40HJC 49797062 IC50 > 100000 nM T15855 CL3P4H 49797063 IC50 > 100000 nM T15855 CPC76U 49797064 IC50 = 55000 nM T15855 C5F4JN 49797065 IC50 = 57000 nM T15855 C86HND 49797066 IC50 = 74000 nM T15855 C8E4XD 49797067 IC50 > 100000 nM T15855 CHO1U0 49797068 IC50 = 39000 nM T15855 CO1TW7 49797069 IC50 > 100000 nM T15855 CAD6W1 49797071 IC50 = 17000 nM T15855 CQYU80 49797072 IC50 > 100000 nM T15855 CEZ38H 49797073 IC50 > 100000 nM T15855 C0CEU7 49797074 IC50 > 100000 nM T15855 C72JXY 49797075 IC50 > 100000 nM T15855 COA41Q 49797076 IC50 = 64000 nM T15855 CPQ3Z2 49797077 IC50 = 58000 nM T15855 C1WI0D 49797078 IC50 = 42000 nM T15855 C4D8XP 49797079 IC50 = 77000 nM T15855 CQG4J6 49797080 IC50 > 100000 nM T15855 CKM9S4 49797081 IC50 > 100000 nM T15855 C3JRW0 49797082 IC50 > 100000 nM T15855 C27IEB 49797083 IC50 > 100000 nM T15855 C0JUL3 49797084 IC50 = 23000 nM T15855 C85DOL 49797085 IC50 > 100000 nM T15855 CEGO30 49797086 IC50 > 100000 nM T15855 C2TC3I 49797087 IC50 > 100000 nM T15855 C04JWY 49797088 IC50 = 9800 nM T15855 CA2U4Y 49797089 IC50 > 100000 nM T15855 CFT46J 49797090 IC50 > 100000 nM T15855 C35TFW 49797091 IC50 > 100000 nM T15855 CRL7Z5 49797092 IC50 > 100000 nM T15855 CYU74X 49797093 IC50 > 100000 nM T15855 C2O3SG 49797094 IC50 > 100000 nM T15855 CFL3O2 49797106 IC50 > 100000 nM T15855 CF4NR7 49797107 IC50 > 100000 nM T15855 CV9QW6 49797108 IC50 > 100000 nM T15855 CJZA65 49797109 IC50 > 100000 nM T15855 CBS36X 49797110 IC50 > 100000 nM T15855 C0STP5 49797111 IC50 > 100000 nM T15855 C7KV5R 49797112 IC50 > 100000 nM T15855 CJPX53 49797113 IC50 > 100000 nM T15855 C2OI0Y 49797114 IC50 > 100000 nM T15855 CW20FJ 49797115 IC50 > 100000 nM T15855 C9P6VU 49797116 IC50 = 41300 nM T15855 C67SIA 49797117 IC50 > 100000 nM T15855 CCI8Y0 49797118 IC50 > 100000 nM T15855 CE10UF 49797119 IC50 > 100000 nM T15855 CLH0V3 49797120 IC50 > 100000 nM T15855 C2N8WX 49797121 IC50 > 100000 nM T15855 CNCE06 49797122 IC50 > 100000 nM T15855 C76UAB 49797123 IC50 > 100000 nM T15855 CHWT89 49797124 IC50 > 100000 nM T15855 C1Z6NE 49797125 IC50 > 100000 nM T15855 C25MQG 49797126 IC50 > 100000 nM T15855 COL54B 49797127 IC50 > 100000 nM T15855 C5OUQ3 49797128 IC50 > 100000 nM T15855 C3NMI8 49797173 Ki = 310 nM T15855 C1E3YB 49797174 Ki = 230 nM T15855 CVD0I1 49797175 Ki = 560 nM T15855 CH02OC 49797176 Ki = 8800 nM T15855 CY1OJ5 49797177 Ki > 30000 nM T15855 C25ZSD 49797191 IC50 > 100000 nM T15855 C0OJX9 49797192 IC50 > 100000 nM T15855 C7GZ4B 49797193 IC50 > 100000 nM T15855 CVT2E5 49797194 IC50 > 100000 nM T15855 C75MGE 49797195 IC50 > 100000 nM T15855 CVS70C 49797196 IC50 > 100000 nM T15855 C42QPW 49797197 IC50 > 100000 nM T15855 C6ZGL5 49797198 IC50 > 100000 nM T15855 C1B5NH 49797199 IC50 > 100000 nM T15855 CGQN24 49797200 IC50 > 100000 nM T15855 CS2AI5 49797201 IC50 > 100000 nM T15855 CM7RE3 49797202 IC50 > 100000 nM T15855 CGM9E7 49797203 IC50 > 100000 nM T15855 COU0I6 49797204 IC50 > 100000 nM T15855 C3XML2 49797205 IC50 > 100000 nM T15855 CP0O2F 49797223 IC50 = 33000 nM T15855 CTH7I8 49797224 IC50 = 34000 nM T15855 CG9P7O 49797225 IC50 = 54000 nM T15855 C3A2QK 49797226 IC50 = 43000 nM T15855 C4NOK2 49797227 IC50 > 100000 nM T15855 CB13PO 49797228 IC50 = 7600 nM T15855 C47VOG 49797229 IC50 > 100000 nM T15855 CD2CL1 49797230 IC50 > 100000 nM T15855 C0LK6B 49797231 IC50 = 5800 nM T15855 CON0A6 49797232 IC50 = 60000 nM T15855 C4AVU3 49797233 IC50 = 33000 nM T15855 CQ93MI 49797234 IC50 = 76000 nM T15855 CO2JV8 49797235 IC50 = 40000 nM T15855 C27LDC 49797236 IC50 = 10000 nM T15855 CA5GM6 49797237 IC50 > 100000 nM T15855 CT8PW1 49797238 IC50 = 25000 nM T15855 CJQ38S 49797239 IC50 = 10000 nM T15855 CT65MR 49797240 IC50 = 66000 nM T15855 C08IFZ 49797241 IC50 > 100000 nM T15855 CA4E8M 49797242 IC50 = 54000 nM T15855 CN8FR2 49797243 IC50 = 49000 nM T15855 C37MDP 49797244 IC50 > 100000 nM T15855 CM41RN 49797245 IC50 > 100000 nM T15855 C59JEK 49797246 IC50 = 28000 nM T15855 CUMH43 49797248 IC50 > 100000 nM T15855 CM59PE 49797249 IC50 > 100000 nM T15855 CN5K1S 49797250 IC50 > 100000 nM T15855 CT5HY0 49797251 IC50 > 100000 nM T15855 C0E5PY 49797252 IC50 > 100000 nM T15855 C3E5JB 49797253 IC50 = 40000 nM T15855 CA8P5N 49797344 IC50 > 100000 nM T15855 CJL2B8 49797345 IC50 > 100000 nM T15855 CT79YI 49797346 IC50 > 100000 nM T15855 C93VJO 49797347 IC50 > 100000 nM T15855 CDI52A 49797348 IC50 > 100000 nM T15855 C7ATK9 49797349 IC50 = 60000 nM T15855 C2Y3DS 49797350 IC50 = 82000 nM T15855 CA4CE3 49797351 IC50 > 100000 nM T15855 C3A8YT 49797352 IC50 > 100000 nM T15855 C1Z8HB 49797353 IC50 = 990 nM T15855 CC0T8H 49797354 IC50 > 100000 nM T15855 C92QND 49797355 IC50 = 21000 nM T15855 C2HPE8 49797356 IC50 > 100000 nM T15855 C9UXH2 49797357 IC50 = 11000 nM T15855 CTYO37 49797358 IC50 > 100000 nM T15855 C1K4FR 49797359 IC50 = 6300 nM T15855 CJ2D0P 49797360 IC50 = 29000 nM T15855 CA3Q2W 49797361 IC50 > 100000 nM T15855 CNMF62 49797362 IC50 = 12000 nM T15855 CLVF17 49797501 IC50 = 11000 nM T15855 CR0AK2 49797502 IC50 = 7900 nM T15855 CM1Y7K 49797503 IC50 = 5300 nM T15855 CUSI73 49797504 IC50 = 3900 nM T15855 CJ0DX6 49797505 IC50 = 5500 nM T15855 C2A7LE 49797506 IC50 = 12000 nM T15855 CU4M3T 49797507 IC50 = 2700 nM T15855 C8GCS5 49797508 IC50 = 4900 nM T15855 CTP9L2 49797509 IC50 = 2500 nM T15855 CT76PM 49797510 IC50 = 3900 nM T15855 C4K0QT 49797511 IC50 = 980 nM T15855 CLHB50 49797512 IC50 = 1500 nM T15855 CC56FE 49797513 IC50 = 5400 nM T15855 C4T6AB 49797514 IC50 = 2000 nM T15855 C41VHF 49797515 IC50 = 17000 nM T15855 CBD9H2 49797516 IC50 = 10000 nM T15855 CAOC90 49797517 IC50 = 6200 nM T15855 C0F5QX 49797518 IC50 = 1900 nM T15855 C7T5XW 49797519 IC50 = 1000 nM T15855 CM6SF5 49797520 IC50 = 1200 nM T15855 CQZN45 49797521 IC50 = 15000 nM T15855 CG64BU 49797522 IC50 = 11000 nM T15855 C5G3MA 49797524 IC50 = 830 nM T15855 CO42DE 49797525 IC50 = 1200 nM T15855 C5L1EP 49797526 IC50 = 1000 nM T15855 CTWR80 49797527 IC50 = 2500 nM T15855 CPIC42 49797528 IC50 = 7200 nM T15855 C5N1ZB 49797529 IC50 = 5700 nM T15855 CU72EZ 49797596 IC50 > 100000 nM T15855 C6AZ2C 49797599 IC50 > 100000 nM T15855 CR86PO 49797604 IC50 > 100000 nM T15855 C6DJX7 49797605 IC50 > 100000 nM T15855 CK3ZI1 49797607 IC50 > 100000 nM T15855 C7AD0C 49797610 IC50 = 45000 nM T15855 C4XHO5 49797612 IC50 > 100000 nM T15855 C7VL5U 49797614 IC50 > 100000 nM T15855 CY09JE 49797615 IC50 > 100000 nM T15855 C1ZLF0 49797616 IC50 > 100000 nM T15855 CN48OE 49797627 IC50 > 100000 nM T15855 CV6I0O 49797630 IC50 > 100000 nM T15855 CAG1U7 49797631 IC50 > 100000 nM T15855 C8JNU1 49797636 IC50 > 100000 nM T15855 C0DN5G 49797642 IC50 > 100000 nM T15855 CJVS96 49797644 IC50 > 100000 nM T15855 CBRT78 49797650 IC50 = 53000 nM T15855 CZW93Y 49797653 IC50 > 100000 nM T15855 COM5Q7 49836030 IC50 > 10000 nM T15855 CKZJ30 49837952 Ki = 33000 nM T15855 CXR05H 49837954 Ki = 39000 nM T15855 C4QSP1 49837961 Ki = 66000 nM T15855 CTDR85 49862539 Ki > 30000 nM T15855 CT8Q9N 49862713 Ki > 30000 nM T15855 C0OB8C 49862714 Ki > 30000 nM T15855 CJ58AG 49862715 Ki > 10000 nM T15855 CPU7F6 49862790 Ki > 30000 nM T15855 C4FZY2 49862791 Ki > 30000 nM T15855 CF40YM 49862792 Ki > 30000 nM T15855 CK0GC5 49864113 Ki = 0.086 nM T15855 CK1CD3 50925423 IC50 > 10000 nM T15855 C7T6PI 50994092 IC50 > 30000 nM T15855 C67CTP 51032641 IC50 > 25000 nM T15855 CL4S9Y 51050450 IC50 > 30000 nM T15855 CLU39H 51051131 IC50 = 11000 nM T15855 C5PRF8 51051132 IC50 = 12000 nM T15855 CYF04M 51051134 IC50 = 820 nM T15855 CPCY75 51051136 IC50 = 630 nM T15855 C7JM3I 51051236 IC50 = 2300 nM T15855 CZ5HJ0 51051238 IC50 = 420 nM T15855 C1OUG5 51051240 IC50 = 2000 nM T15855 C6GAP9 51051329 IC50 > 30000 nM T15855 C9KPJ6 51051331 IC50 > 100000 nM T15855 C85CEJ 51346970 IC50 > 100000 nM T15855 C4PFT3 51346971 IC50 > 100000 nM T15855 CLND76 51356956 Ki = 25000 nM T15855 CH92AI 51356957 Ki = 106000 nM T15855 CH89VX 51356958 Ki = 137000 nM T15855 C5D4HV 51356959 Ki = 179000 nM T15855 C8WOG2 51356962 Ki = 182000 nM T15855 C4VC2U 52942435 IC50 > 10000 nM T15855 C2B6EX 52943488 Ki > 10000 nM T15855 C56CXU 52943631 IC50 > 10000 nM T15855 CHD7O6 52943758 IC50 > 10000 nM T15855 C4I6ML 52944843 IC50 > 10000 nM T15855 C57XSM 52944845 IC50 > 10000 nM T15855 CT6SQ3 52944941 IC50 > 10000 nM T15855 C7RJM9 52945660 IC50 = 360 nM T15855 C9OAF1 52946149 IC50 > 10000 nM T15855 CC56BV 52946866 IC50 > 100000 nM T15855 CC7N8S 52948914 IC50 > 10000 nM T15855 C4LVO6 52948971 IC50 > 10000 nM T15855 CTU0J1 52949742 IC50 > 10000 nM T15855 CD4HQ1 53233695 IC50 > 30000 nM T15855 C89KWN 53233798 IC50 = 11000 nM T15855 CEFX05 53311069 IC50 > 100000 nM T15855 CQL50R 53311070 IC50 > 100000 nM T15855 C1Q4WK 53311071 IC50 > 100000 nM T15855 C67LHZ 53311072 IC50 > 100000 nM T15855 CQ0ZJ2 53311073 IC50 > 100000 nM T15855 C7PMY1 53311074 IC50 > 100000 nM T15855 CWN9H7 53311140 IC50 > 100000 nM T15855 CAL51C 53311141 IC50 > 100000 nM T15855 C2SXV0 53311142 IC50 > 100000 nM T15855 C7AEF8 53311143 IC50 > 100000 nM T15855 C5IOZ6 53311144 IC50 > 100000 nM T15855 CVR4H3 53311222 IC50 > 100000 nM T15855 CNX08H 53311223 IC50 > 100000 nM T15855 CET6W5 53311225 IC50 > 100000 nM T15855 C3RZS4 53311226 IC50 > 100000 nM T15855 CHR17Y 53311227 IC50 > 100000 nM T15855 C3HGW8 53312238 IC50 > 100000 nM T15855 CM03UX 53312239 IC50 > 100000 nM T15855 C9K4CZ 53312243 IC50 > 100000 nM T15855 CU4BS2 53312323 IC50 > 100000 nM T15855 CF5I6O 53312326 IC50 > 100000 nM T15855 C6PSL2 53312327 IC50 > 100000 nM T15855 C0WYS5 53312328 IC50 > 100000 nM T15855 CYC69Q 53317564 IC50 > 69000 nM T15855 C0QOV9 53317565 IC50 > 100000 nM T15855 CURC70 53317566 IC50 > 100000 nM T15855 C3ZK1W 53317575 IC50 = 5800 nM T15855 CBQ0J7 53317579 IC50 = 10000 nM T15855 CIY9F7 53317580 IC50 = 14000 nM T15855 C5DMS9 53317581 IC50 > 100000 nM T15855 C1XD9W 53317582 IC50 = 37000 nM T15855 CR0O8T 53317583 IC50 = 18000 nM T15855 C9GLH7 53318841 IC50 = 65000 nM T15855 C06TDE 53318842 IC50 = 55000 nM T15855 C73TER 53318856 IC50 > 100000 nM T15855 CC56NE 53318863 IC50 > 100000 nM T15855 C4UJI8 53318864 IC50 = 58000 nM T15855 C8CZ2A 53318865 IC50 = 32000 nM T15855 CLVY47 53318866 IC50 = 72000 nM T15855 CM7S5W 53319067 IC50 = 30000 nM T15855 C1X3NE 53320178 IC50 = 70000 nM T15855 C1P8BK 53320179 IC50 = 35000 nM T15855 C50UBZ 53320180 IC50 > 100000 nM T15855 C2JTR7 53320181 IC50 > 100000 nM T15855 C0TYJ5 53320182 IC50 = 46000 nM T15855 C7RSX2 53320183 IC50 = 26000 nM T15855 C9XGE4 53321472 IC50 = 69000 nM T15855 CY0ZV9 53321485 IC50 > 100000 nM T15855 CK0OB2 53321486 IC50 > 100000 nM T15855 CNK34J 53321487 IC50 > 100000 nM T15855 C7EO3D 53321495 IC50 = 58000 nM T15855 C3M7PQ 53321496 IC50 = 22000 nM T15855 C0NUQ7 53321497 IC50 = 21000 nM T15855 C31DSJ 53321498 IC50 = 29000 nM T15855 C2ZKV9 53321499 IC50 = 19000 nM T15855 CB76JK 53321550 IC50 = 26000 nM T15855 C3QT0R 53321621 IC50 = 61000 nM T15855 CF2GQ1 53321670 IC50 = 25000 nM T15855 CXIS21 53322758 IC50 > 100000 nM T15855 CY71QL 53322814 IC50 > 100000 nM T15855 CLU96Y 53322820 IC50 = 33000 nM T15855 C8YVF1 53322821 IC50 > 100000 nM T15855 C4QS6V 53322822 IC50 > 100000 nM T15855 C62JTB 53322823 IC50 = 76000 nM T15855 CT14FU 53322824 IC50 > 100000 nM T15855 CXJ1F8 53322825 IC50 = 31000 nM T15855 C3K1VY 53322826 IC50 = 58000 nM T15855 C9N6HK 53322952 IC50 > 100000 nM T15855 C9LU8M 53324129 IC50 = 34000 nM T15855 CCY7M0 53324130 IC50 = 76000 nM T15855 C4F1QK 53324142 IC50 > 100000 nM T15855 CZN71C 53324143 IC50 > 100000 nM T15855 CG83JZ 53324144 IC50 > 100000 nM T15855 CE8J1D 53324145 IC50 > 100000 nM T15855 C0Y3AC 53324153 IC50 > 100000 nM T15855 C9O1IW 53324154 IC50 = 75000 nM T15855 CTW5G0 53324155 IC50 = 95000 nM T15855 C2DPZ0 53324156 IC50 = 39000 nM T15855 CL5Z8N 53324211 IC50 = 11400 nM T15855 CV7UM8 53324212 IC50 > 30000 nM T15855 C98EJV 53324213 IC50 > 30000 nM T15855 CSN28M 53324293 IC50 > 100000 nM T15855 C25OJW 53325399 IC50 = 5500 nM T15855 CXW5O9 53325446 IC50 = 71000 nM T15855 C1SO0C 53325447 IC50 > 100000 nM T15855 C1S3WB 53325453 IC50 = 25000 nM T15855 C2KFW6 53325454 IC50 = 35000 nM T15855 C4ZFR5 53325455 IC50 = 47000 nM T15855 CW8TM9 53325504 IC50 > 30000 nM T15855 CV0H8P 53326691 IC50 = 65000 nM T15855 C3ZWN6 53326704 IC50 = 62000 nM T15855 C73SKG 53326705 IC50 > 100000 nM T15855 CG9V4W 53326706 IC50 = 50000 nM T15855 C5K8CP 53326713 IC50 > 100000 nM T15855 CN12AO 53353383 IC50 = 27000 nM T15855 C51GUC 53354365 IC50 = 57000 nM T15855 CRJ5P9 53354369 IC50 > 100000 nM T15855 C4G2HT 53354470 IC50 = 69000 nM T15855 CUC1N3 53356519 Ki = 2238 nM T15855 CSD1Q4 53357353 IC50 > 60000 nM T15855 C5P9VZ 53465973 IC50 = 960 nM T15855 C7OBF2 53465974 IC50 = 4000 nM T15855 CF5YJ8 53465975 IC50 > 10000 nM T15855 C5XER7 53466046 IC50 = 8.8 nM T15855 CJ9T8M 53466047 Ki = 6.5 nM T15855 CP1CL8 53466049 IC50 = 141 nM T15855 CPSQ16 53466050 IC50 = 34800 nM T15855 C4UC1P 53466119 IC50 = 80 nM T15855 C59SML 53466121 IC50 = 80 nM T15855 C7JPY2 53466122 IC50 = 32 nM T15855 CYZK63 53466123 Ki = 37 nM T15855 CVJ0D5 53466193 IC50 = 166 nM T15855 C2XE8Y 53466195 IC50 = 29 nM T15855 C0P2YE 53466196 IC50 = 310 nM T15855 CPA0K4 53466271 IC50 = 730 nM T15855 CYG36O 53466361 IC50 = 1100 nM T15855 C0ZQ5T 54581616 IC50 = 21000 nM T15855 C5UW0D 56652661 IC50 > 100000 nM T15855 C1QX0O 56657809 IC50 = 53000 nM T15855 CU74VH 56658024 IC50 = 6800 nM T15855 CF6PV5 56658026 IC50 = 910 nM T15855 C2KI8Y 56658028 IC50 = 9400 nM T15855 CY4E6U 56658138 IC50 > 10000 nM T15855 C1PI4L 56664962 IC50 = 4500 nM T15855 CXH5W7 56671896 IC50 = 278 nM T15855 CBK31U 56675279 IC50 = 3910 nM T15855 CW8KU6 56675536 IC50 = 9.4 nM T15855 C9OL5C 56962798 IC50 > 100000 nM T15855 CQX8J0 57385070 IC50 > 25000 nM T15855 CPS89B 57385071 IC50 > 25000 nM T15855 CNU9C0 57385072 IC50 > 10000 nM T15855 CG5MT6 57385073 IC50 > 10000 nM T15855 CQZ09L 57390626 IC50 > 100 nM T15855 CWR4E5 57390923 Ki = 993 nM T15855 C0RAD8 57390924 Ki = 802 nM T15855 C5U6RF 57392407 IC50 = 76 nM T15855 CD0OT2 57392409 IC50 > 100 nM T15855 C4QYJ6 57392724 Ki = 2688 nM T15855 CWDY79 57394441 Ki = 3701 nM T15855 CZ23RJ 57395915 IC50 > 100 nM T15855 C8KMS2 57396206 Ki = 60 nM T15855 C2QL6K 57397702 IC50 = 58 nM T15855 CBQ85O 57397704 IC50 = 43 nM T15855 C2ZE3R 57397706 IC50 = 12 nM T15855 CW97SN 57398006 Ki = 1894 nM T15855 C01KCU 57399665 Ki = 967 nM T15855 C65ZFW 57401128 IC50 = 45 nM T15855 CYX43T 57401419 Ki = 3477 nM T15855 C1T0AD 57403169 Ki = 823 nM T15855 C12QCM 57403170 Ki = 3106 nM T15855 CX94UQ 57403171 Ki = 558 nM T15855 C1L8YD 57404359 IC50 = 2260 nM T15855 C8SX7A 57404360 IC50 = 2600 nM T15855 C0Q1OZ 57404374 IC50 > 50000 nM T15855 CL0UA1 57525787 IC50 = 72.4 nM T15855 C9ZE7J 58874273 IC50 > 100000 nM T15855 CZ4VD5 60032916 IC50 = 9.2 nM T15855 C9SND1 68305755 IC50 > 100000 nM T15855 CP3E2X 68416066 IC50 = 86 nM T15855 CCS6K9 68417211 IC50 = 220 nM T15855 CH3Z7F 68658979 IC50 = 5000 nM T15855 C6HRX1 68845950 IC50 = 45800 nM T15855 CWTN63 69446993 IC50 > 100000 nM T15855 CK26FY 70295607 IC50 > 30000 nM T15855 CV4X5S 70295927 IC50 = 22400 nM T15855 CXSV41 70296244 IC50 = 19400 nM T15855 C3SB1V 70296823 IC50 = 30000 nM T15855 CXD5V6 70297609 IC50 = 7400 nM T15855 CEG1L5 70330884 IC50 = 480 nM T15855 C5W6LY 70681316 IC50 = 33000 nM T15855 C97JFS 70682267 IC50 = 320 nM T15855 CE1FU2 70682268 IC50 = 114 nM T15855 C4YW5T 70684349 IC50 = 510 nM T15855 C6W1CT 70684350 IC50 = 27000 nM T15855 C1GF3E 70684351 IC50 = 17 nM T15855 C1Q3ZO 70686506 IC50 = 5.9 nM T15855 CLQC52 70688610 IC50 = 54 nM T15855 CVYH31 70689717 IC50 = 23000 nM T15855 CYO5X6 70690674 IC50 = 43 nM T15855 C2J7FS 70690675 IC50 = 19 nM T15855 CL6KR9 70690676 IC50 = 1.2 nM T15855 C19FJC 70692822 IC50 = 500 nM T15855 C8JZ3Q 70692823 IC50 = 530 nM T15855 CIX3F9 70694853 IC50 = 110 nM T15855 CQJD92 70694854 IC50 = 27 nM T15855 C1NGL5 70696903 IC50 = 23 nM T15855 C31UTS 71184301 IC50 = 14700 nM T15855 C8LY1U 71184352 IC50 > 30000 nM T15855 C9IRW7 71184590 IC50 = 28300 nM T15855 C08NDK 71184749 IC50 = 10800 nM T15855 CP91OE 71203742 IC50 > 100000 nM T15855 CP6G5W 71203746 IC50 > 100000 nM T15855 C32UMV 71203748 IC50 > 100000 nM T15855 C04XQY 71203752 IC50 > 100000 nM T15855 CE2I0K 71203758 IC50 > 100000 nM T15855 CIQ7O2 71203767 IC50 = 21163 nM T15855 C5GEJ9 71203769 IC50 > 100000 nM T15855 C7LKV0 71203783 IC50 > 100000 nM T15855 CAJ8F0 71449608 IC50 > 10000 nM T15855 CP9K2W 71450603 IC50 = 5000 nM T15855 C61LNR 71452448 IC50 = 13600 nM T15855 CN4FE7 71454208 IC50 = 16000 nM T15855 C1LRH5 71455960 IC50 = 45400 nM T15855 C59TGZ 71457761 IC50 = 4100 nM T15855 C5T6QP 71457765 IC50 = 20900 nM T15855 CUB4V8 71459679 IC50 = 6300 nM T15855 CKZ17B 71463121 IC50 = 9600 nM T15855 C4VKM3 71463122 IC50 = 9200 nM T15855 C8T2PW 71655265 IC50 = 1900 nM T15855 CVB75Q 71655394 IC50 = 1700 nM T15855 CH4ZS0 71655395 IC50 > 100000 nM T15855 C7BD2R 71720854 IC50 = 1200 nM T15855 CW3JG7 71731241 IC50 > 100000 nM T15855 C3D4HJ 71731243 IC50 > 100000 nM T15855 CU6BC5 71731355 IC50 > 100000 nM T15855 C5TS9Y 71731356 IC50 > 100000 nM T15855 C5RTY9 71731357 IC50 > 100000 nM T15855 CD9F5X 71731476 IC50 > 100000 nM T15855 C3IO9H 71731477 IC50 > 100000 nM T15855 CVAD62 71731478 IC50 > 100000 nM T15855 C1ON0X 71731479 IC50 > 100000 nM T15855 CZYQ05 71731604 IC50 > 100000 nM T15855 C40YRO 71731605 IC50 > 100000 nM T15855 C9Q8MO 72164809 IC50 = 680 nM T15855 CL5X1Z 72164811 IC50 = 280 nM T15855 C7N8WB 72164813 IC50 = 1130 nM T15855 C2R0NV 72164815 IC50 = 510 nM T15855 C4JLM5 72164817 IC50 = 330 nM T15855 C6RQ9A 72164819 IC50 = 430 nM T15855 C38GWP 72164942 IC50 = 440 nM T15855 C4T0MY 72164944 IC50 = 390 nM T15855 C0T4UW 72164946 IC50 = 320 nM T15855 CLV02R 72164948 IC50 = 340 nM T15855 CHPN10 72164950 IC50 = 1210 nM T15855 CI78FQ 72165082 IC50 = 300 nM T15855 CN0VU2 72165084 IC50 = 450 nM T15855 C84SYX 72165086 IC50 = 690 nM T15855 C1RQA3 72165088 IC50 = 240 nM T15855 CH51ZR 72165090 IC50 = 470 nM T15855 C1HL2A 72188903 IC50 > 100000 nM T15855 CLS1A0 72188904 IC50 > 100000 nM T15855 CL7P3D 72193502 IC50 > 100000 nM T15855 C4AXB8 72193503 IC50 = 28000 nM T15855 CQC28P 72193504 IC50 > 100000 nM T15855 CV87PE 72193505 IC50 > 100000 nM T15855 C65DFP 72697059 IC50 = 9400 nM T15855 CX07OC 72697060 IC50 = 630 nM T15855 CZ56DO 72697061 IC50 = 6600 nM T15855 C1A2KX 72697062 IC50 = 6220 nM T15855 CS5U1F 72697063 IC50 = 46820 nM T15855 CA3HI1 72697064 IC50 = 520 nM T15855 CCZJ47 72697206 IC50 = 3040 nM T15855 CWNZ91 72697207 IC50 = 7910 nM T15855 C6BWI4 72697208 IC50 = 52120 nM T15855 C9JA1Q 72697209 IC50 = 960 nM T15855 CF6A8N 72697210 IC50 = 900 nM T15855 CTMR03 72697211 IC50 = 2720 nM T15855 CP9NV5 72697212 IC50 = 40770 nM T15855 C1P8HS 72697352 IC50 = 17560 nM T15855 CC7G3M 72697353 IC50 = 29600 nM T15855 CXYO73 72697354 IC50 = 520 nM T15855 CAXV78 72697355 IC50 = 22510 nM T15855 CGV09W 72697356 IC50 = 2910 nM T15855 CIF9D7 72697357 IC50 = 2550 nM T15855 CC8RA6 72697358 IC50 = 1340 nM T15855 C1EC7S 72697359 IC50 > 58000 nM T15855 C8CRO6 72697494 IC50 = 3110 nM T15855 C03NKY 72697495 IC50 = 240 nM T15855 CP0MU3 72697496 IC50 = 7190 nM T15855 CI60AK 72697497 IC50 = 3420 nM T15855 CO19YK 72697498 IC50 = 4940 nM T15855 C47IGZ 72697499 IC50 = 8970 nM T15855 C65OPG 72697500 IC50 = 960 nM T15855 C3ZP7N 72697501 IC50 = 1070 nM T15855 C7EF8C 72697646 IC50 = 2350 nM T15855 C08IGP 72699737 IC50 > 100000 nM T15855 CAEF04 72707536 IC50 > 100000 nM T15855 C7ARW4 72707537 IC50 > 100000 nM T15855 CSZR98 73346173 IC50 > 100000 nM T15855 C1L4RX 73346174 IC50 > 100000 nM T15855 CGNL10 73347698 IC50 > 100000 nM T15855 CO5TB8 73349220 IC50 = 50000 nM T15855 CNC6B8 73350798 IC50 = 39000 nM T15855 CDBV29 73350799 IC50 > 100000 nM T15855 CYG04J 73352283 IC50 > 100000 nM T15855 CV6BA3 73353756 IC50 > 100000 nM T15855 C51QGP 73353757 IC50 > 100000 nM T15855 CBK37N 73353758 IC50 > 100000 nM T15855 CLO76J 73355285 IC50 > 100000 nM T15855 CCVT96 73355286 IC50 = 220 nM T15855 CY0N9K 76311138 IC50 = 55700 nM T15855 CWK7M6 76311139 IC50 = 1000 nM T15855 CIP4R0 76314754 IC50 = 3300 nM T15855 C3HRA1 76314755 IC50 = 1300 nM T15855 C68JOX 76318341 IC50 = 12300 nM T15855 CET31O 76318342 IC50 = 1800 nM T15855 C9UGA3 76325642 IC50 > 288200 nM T15855 CNIP02 76325643 IC50 = 1400 nM T15855 C08DYM 76325644 IC50 = 700 nM T15855 C3C7HE 76325645 IC50 = 4700 nM T15855 CW4M6E 76329221 IC50 = 900 nM T15855 CH95ZJ 76336484 IC50 = 125100 nM T15855 CTXI04 86267501 IC50 > 10000 nM T15855 CO78UK 86267502 IC50 > 10000 nM T15855 CLG83C 86268944 IC50 > 10000 nM T15855 C31OGJ 86279928 IC50 > 10000 nM T15855 CB60OP 89488720 IC50 > 100000 nM T15855 CU9LB2 90664438 IC50 = 230 nM T15855 CQ20XA 90664578 IC50 = 15900 nM T15855 CV87ZH 90664579 IC50 = 63 nM T15855 CDEN13 90664693 IC50 = 520 nM T15855 CV0SF5 90664925 IC50 > 100000 nM T15855 CBQ38C 101879512 IC50 = 56330 nM T15855 CZ1G3O 118712516 IC50 > 100000 nM T15855 C8X4JA 118712517 IC50 > 100000 nM T15855 CC29AB 118712518 IC50 > 100000 nM T15855 CB09PD 118712519 IC50 > 100000 nM T15855 CD4U1X 118712520 IC50 > 100000 nM T15855 CU0V5J 118712521 IC50 > 100000 nM T15855 C03OUP 118712522 IC50 > 100000 nM T15855 CT2MZ8 118712764 IC50 = 600 nM T15855 C3W5RU 118712765 IC50 = 490 nM T15855 CKA1N5 118712766 IC50 = 710 nM T15855 C8M6ZW 118712767 IC50 = 1050 nM T15855 CV5C6D 118712768 IC50 = 680 nM T15855 C2NSC7 118712769 IC50 = 640 nM T15855 CAR4W5 118712772 IC50 = 670 nM T15855 CRWT85 118712773 IC50 = 190 nM T15855 C4T2FY 118712775 IC50 = 1010 nM T15855 CJ8EL0 118712778 IC50 = 5690 nM T15855 C07UOL 118712779 IC50 = 76720 nM T15855 C25HYG 118712780 IC50 = 36530 nM T15855 CD0HQ4 118712781 IC50 = 51600 nM T15855 C46TMQ 118712785 IC50 = 2120 nM T15855 C5M3BX 118712788 IC50 = 8980 nM T15855 CK7HN4 118722408 IC50 = 3420 nM T15855 CK71WT 118722410 IC50 = 750 nM T15855 CI74ZM 118722411 IC50 = 880 nM T15855 CH1P7Y 118722412 IC50 = 1750 nM T15855 CL8TY5 118722413 IC50 = 4170 nM T15855 C8KUP0 118722416 IC50 = 1470 nM T15855 COG4V6 118722421 IC50 = 2900 nM T15855 C7TEY3 122178433 IC50 > 10000 nM T15855 C6PLX9 127035081 IC50 = 44000 nM T15855 CJ0KS7 127035239 IC50 > 100000 nM T15855 CKSZ13 127035240 IC50 > 100000 nM T15855 C6T1IM 127035241 IC50 > 100000 nM T15855 CJRL72 127035242 IC50 > 100000 nM T15855 CVKI59 127035243 IC50 = 41000 nM T15855 CWJX95 127035244 IC50 = 25000 nM T15855 C0XMS7 127035375 IC50 = 27000 nM T15855 CMK5Q9 127035376 IC50 > 100000 nM T15855 C4N7QB 127035377 IC50 > 100000 nM T15855 CGN49F 127035378 IC50 = 55000 nM T15855 C36UHW 127035569 IC50 = 62000 nM T15855 CTKS36 127035740 IC50 = 47000 nM T15855 CAXT02 127035741 IC50 > 100000 nM T15855 CZB0L6 127035742 IC50 = 89000 nM T15855 C4QWL5 127035743 IC50 > 100000 nM T15855 CPGF39 127035744 IC50 = 91000 nM T15855 CXTD34 127035745 IC50 > 100000 nM T15855 CM98XR 127035752 IC50 = 60000 nM T15855 C87MVA 127035753 IC50 > 100000 nM T15855 CDW25O 127035754 IC50 = 41000 nM T15855 CN08IS 127045827 IC50 > 100000 nM T15855 CAK85G 127046590 IC50 = 7090 nM T15855 CP3U8J 127046622 IC50 = 370 nM T15855 CFAI71 127046624 IC50 = 10000 nM T15855 CB6PA7 127046626 IC50 = 3700 nM T15855 C76IGF 127046628 IC50 > 25000 nM T15855 CHL49F 127046630 IC50 = 36 nM T15855 CH0D2Z 127046632 IC50 = 4700 nM T15855 CK4SO7 127047730 IC50 = 17 nM T15855 CSO9L3 127047731 IC50 = 37 nM T15855 C4KIA9 127047732 IC50 = 1700 nM T15855 CHX41E 127047733 IC50 = 119 nM T15855 C6I7HW 127047734 IC50 = 113 nM T15855 C2CP4F 127047761 IC50 = 50 nM T15855 CYR1X2 127047762 IC50 > 100000 nM T15855 CIV4C2 127047839 IC50 = 80 nM T15855 CDYA70 127047985 IC50 = 1980 nM T15855 C0FS5E 127048116 IC50 = 550 nM T15855 C6NIM5 127048874 IC50 = 34000 nM T15855 CXD69M 127048875 IC50 = 36000 nM T15855 C65MAC 127048876 IC50 = 100000 nM T15855 C23BWQ 127049179 IC50 = 100000 nM T15855 CNCB06 127049180 IC50 = 46000 nM T15855 CJ8SG3 127049204 IC50 = 59000 nM T15855 CRM04V 127049507 IC50 = 100000 nM T15855 C76VPA 127049823 IC50 = 50000 nM T15855 CH0X6Q 127050132 IC50 = 100000 nM T15855 CIGA32 127050759 IC50 = 41000 nM T15855 CNY90B 127050760 IC50 = 100000 nM T15855 C80WCY 127050761 IC50 = 100000 nM T15855 CUVQ34 127050762 IC50 = 100000 nM T15855 CJMS57 127051032 IC50 = 18000 nM T15855 C9V4EG 127051045 IC50 = 37000 nM T15855 C7W8JR 127051639 IC50 = 79000 nM T15855 C36SXH 127052286 IC50 = 63000 nM T15855 CBR1F8 127052287 IC50 = 20000 nM T15855 CHZX75 127052288 IC50 = 19000 nM T15855 CB34GQ 127052289 IC50 = 100000 nM T15855 CLG0Q3 127052290 IC50 = 43000 nM T15855 CL2S0F 127052581 IC50 = 34000 nM T15855 C1W5AL 127052582 IC50 = 42000 nM T15855 C4TI8H 127052590 IC50 = 65000 nM T15855 CNV0A8 127052636 IC50 = 8100 nM T15855 CS2Z9R 127052637 IC50 = 8000 nM T15855 C75EAL 127052638 IC50 = 3000 nM T15855 CRM4Q8 135518358 IC50 > 100000 nM T15855 CMI5A6 135964368 IC50 = 47000 nM T15855 CO04QA 136177302 IC50 = 80000 nM T15855 CR4VI2 137225025 IC50 = 92000 nM T15855 C3SKH4 145948172 IC50 = 30000 nM T15855 CR9S6F 145958227 IC50 > 300000 nM T15855 CBL76R 145964231 IC50 > 100000 nM T15855 CF53NA 145964407 IC50 > 100000 nM T15855 CNMT16 145965136 IC50 > 100000 nM T15855 CP7VT2 145973710 IC50 > 100000 nM T15855 C9C4WU 145975568 IC50 > 100000 nM T15855 CWF4Y7 145977953 IC50 > 100000 nM T15855 CR3I9D 145978547 IC50 > 100000 nM T15855 CM6L4K 155510749 IC50 > 100000 nM T15855 C5ZQ7W 155511281 IC50 > 100000 nM T15855 CQA73O 155512586 IC50 > 100000 nM T15855 C57QZJ 155512836 IC50 > 100000 nM T15855 CX3U8Z 155515016 IC50 > 100000 nM T15855 C19ZCJ 155518265 IC50 > 100000 nM T15855 C8UOJ4 155518381 IC50 > 100000 nM T15855 CW0NI8 155519444 IC50 > 100000 nM T15855 C3I8AW 155520161 IC50 > 100000 nM T15855 C4AZ9V 155523785 IC50 > 100000 nM T15855 CTSA30 155526359 IC50 > 100000 nM T15855 CVD89H 155526728 IC50 > 100000 nM T15855 C5C4UV 155526759 IC50 > 100000 nM T15855 CAT3J0 155526949 IC50 > 100000 nM T15855 CLE9I0 155528648 IC50 > 100000 nM T15855 C8FHJ2 155529886 IC50 > 100000 nM T15855 CCX9H6 155530472 IC50 > 100000 nM T15855 CB6N4S 155531120 IC50 > 100000 nM T15855 CGV6C1 155531169 IC50 > 100000 nM T15855 CEOQ32 155531330 IC50 > 100000 nM T15855 CN04KW 155533304 IC50 > 100000 nM T15855 CG3RS6 155540249 IC50 > 100000 nM T15855 CJ67GL 155540375 IC50 > 100000 nM T15855 CY25EZ 155544299 IC50 > 100000 nM T15855 C8H3MJ 155544665 IC50 > 100000 nM T15855 CU17DA 155544967 IC50 > 100000 nM T15855 C62YMT 155545522 IC50 > 100000 nM T15855 CNA9X4 155548276 IC50 > 100000 nM T15855 CM9K4B 155548792 IC50 > 100000 nM T15855 CB1AF4 155549522 IC50 > 100000 nM T15855 CX9Y4B 155552378 IC50 > 100000 nM T15855 C1D5QZ 155554658 IC50 > 100000 nM T15855 C7KVR5 155559306 IC50 > 100000 nM T15855 C68CRH 155561682 IC50 > 100000 nM T15855 C48ETF 155565121 IC50 > 100000 nM T15855 CI5C6P 155568161 IC50 > 100000 nM T15855 CUQL05 155568269 IC50 > 100000 nM T15855 D02RDY 11375559 IC50 = 14 nM T15855 D03DNV 71655266 IC50 = 5600 nM T15855 D04CAR 10607286 Ki = 3.1 nM T15855 D07ALM 11232124 IC50 = 142000 nM T15855 D07IJU 13578534 IC50 = 50000 nM T15855 D08NMS 46900258 Ki = 0.27 nM T15855 D0CP1J 56658139 IC50 = 12 nM T15855 D0L9XR 447256 IC50 = 5200 nM T15855 D0N1FU 6918465 IC50 = 6000 nM T15855 D0N1QQ 94701 Ki = 39000 nM T15855 D0R5OE 44422449 IC50 = 4687 nM T15855 D0T2EW 11075394 IC50 = 27 nM T15855 D0Y5IQ 44255320 IC50 = 10000 nM T63609 D02UOZ 2815031 IC50 = 10000 nM T63609 D0Y7VM 47936 EC50 = 500 nM T63609 C4G1YQ 867466 IC50 = 2300 nM T63609 CYJT36 2057741 IC50 = 16000 nM T63609 CUR0M9 2104512 IC50 = 9900 nM T63609 CK3I7Q 3292510 IC50 = 1600 nM T63609 CV7Z3S 3329455 IC50 = 7500 nM T63609 C7D4AU 3409080 IC50 = 13000 nM T63609 C1WPX9 3409372 IC50 = 6400 nM T63609 C3GJT1 3437957 IC50 = 11000 nM T63609 COM4U0 3516249 IC50 = 3100 nM T63609 C4Z2YH 3560838 IC50 = 5300 nM T63609 CZR0I9 3612751 IC50 = 10000 nM T63609 CK1XC3 4106253 IC50 = 10000 nM T63609 CX80GS 4119545 IC50 = 9600 nM T63609 CGM76I 4123757 IC50 = 12000 nM T63609 CXU18Z 4128171 IC50 = 8900 nM T63609 C4R9WU 4133481 IC50 = 15000 nM T63609 CWYM24 4141139 IC50 = 3400 nM T63609 CIG04X 4176698 IC50 = 1000 nM T63609 CV1R6S 4186096 IC50 = 1500 nM T63609 CV47LC 4252177 IC50 = 17000 nM T63609 C07QTY 4258374 IC50 = 5400 nM T63609 C3UQ4G 4287546 IC50 = 5100 nM T63609 C7EF1V 4296739 IC50 = 13000 nM T63609 CE3X6R 4392265 IC50 = 31000 nM T63609 CS72QU 4418394 IC50 = 5900 nM T63609 C5UOW9 4451500 IC50 = 28000 nM T63609 C6CV0J 4456704 IC50 = 6500 nM T63609 CJGR73 4461060 IC50 = 4200 nM T63609 CH2Z5J 4464310 IC50 = 5000 nM T63609 C8BY1K 4591135 IC50 = 3400 nM T63609 CLSY63 4986173 IC50 = 29000 nM T63609 CME82Y 5048573 IC50 = 7300 nM T63609 CFLV26 5050383 IC50 = 7700 nM T63609 CZC82V 5076360 IC50 = 15000 nM T63609 CG31FS 5111500 IC50 = 2800 nM T63609 C12BGF 5111944 IC50 = 4600 nM T63609 CLZY58 5215090 IC50 = 3400 nM T63609 CN94IF 7266923 IC50 = 11000 nM T63609 CDQ3F8 7266928 IC50 = 1700 nM T63609 CMH06Z 7565269 IC50 = 9500 nM T63609 CY1F4E 10072678 IC50 < 150 nM T63609 C5GP9D 10097750 IC50 > 150 nM T63609 CT3XJ9 10505406 IC50 < 150 nM T63609 CAK6E7 10505800 EC50 = 1000 nM T63609 CF94JK 10527678 IC50 = 555 nM T63609 C98VYJ 10527709 IC50 = 192 nM T63609 CTKI14 10529681 IC50 > 150 nM T63609 C7PM6A 10529872 EC50 = 1100 nM T63609 CW0CN8 10553891 IC50 = 251 nM T63609 C4W8OX 10554961 IC50 < 150 nM T63609 C50QUC 10575591 EC50 > 2000 nM T63609 C9W6KY 10576774 IC50 = 228 nM T63609 C0C3OQ 10577997 EC50 < 2000 nM T63609 CE7R3V 10578148 IC50 < 150 nM T63609 CSJQ49 10578739 IC50 = 36 nM T63609 C2CJR0 10601356 IC50 < 150 nM T63609 C4JFR7 10602105 IC50 = 123 nM T63609 C75VJM 10624162 IC50 = 318 nM T63609 CG25XM 10626914 IC50 < 150 nM T63609 C20EOH 10649543 IC50 = 117 nM T63609 CNU40T 10649691 IC50 = 184 nM T63609 C7OI0F 10650063 IC50 > 150 nM T63609 C3IMP1 10694983 IC50 < 150 nM T63609 CDU71E 10695573 IC50 < 150 nM T63609 CDT57L 10719964 IC50 < 150 nM T63609 C7U6WA 10720052 IC50 = 680 nM T63609 C85YXL 10720524 IC50 = 185 nM T63609 CLZJ03 10720525 IC50 < 150 nM T63609 C61BUL 10742236 IC50 = 157 nM T63609 CCV8G1 10742399 IC50 = 43 nM T63609 C6Q3YH 10743405 IC50 = 247 nM T63609 CLV26X 10744316 IC50 > 150 nM T63609 CZP2B5 10745417 IC50 = 21 nM T63609 CXCD37 10768166 IC50 = 65 nM T63609 C2K5HA 10768558 IC50 = 162 nM T63609 CJ4N6I 10769003 IC50 = 117 nM T63609 CUCT02 10792834 IC50 < 150 nM T63609 CI1LR2 10837986 EC50 > 2000 nM T63609 C61ZYI 10838058 EC50 = 1600 nM T63609 C9Z1UP 10838963 EC50 > 2000 nM T63609 CU6RM4 14563677 IC50 > 150 nM T63609 C0AI3P 14788226 Ki > 5000 nM T63609 C0ZNC3 15098733 IC50 < 150 nM T63609 CBQ3Y2 15098745 IC50 = 31 nM T63609 CHA9O8 40957319 IC50 = 11000 nM T63609 CRGS16 41709643 IC50 = 25000 nM T63609 CD0O3R 41709650 IC50 = 16000 nM T63609 CIL67P 41709652 IC50 = 14000 nM T63609 CR04UW 41709679 IC50 = 13000 nM T63609 C79UKE 41709683 IC50 = 11000 nM T63609 CDK09H 41709689 IC50 = 8600 nM T63609 C2G1NF 41709709 IC50 = 22000 nM T63609 CFHP67 41709770 IC50 = 6000 nM T63609 CQ9J4R 41709784 IC50 = 8100 nM T63609 C4T1IY 41709944 IC50 = 10000 nM T63609 C9TKM3 41710028 IC50 = 6600 nM T63609 C4X0VF 44325532 IC50 = 236 nM T63609 CI32AY 137370439 IC50 = 1400 nM T63609 CD59OF 137370506 IC50 = 5000 nM T63609 C04MZR 137370522 IC50 = 1400 nM T63609 C2W8AC 137370592 IC50 = 1200 nM T63609 C75RTL 137370598 IC50 = 26000 nM T63609 CNM96L 137370624 IC50 = 2300 nM T63609 C6HX5O 137370637 IC50 = 9600 nM T63609 CUG19I 137370659 IC50 = 4800 nM T63609 C9Q6HU 137370739 IC50 = 7300 nM T63609 CEW89V 137370768 IC50 = 3700 nM T63609 CDO6E8 137370816 IC50 = 9400 nM T63609 C0D8VK 137370858 IC50 = 4600 nM T63609 C5DL6C 137370883 IC50 = 9100 nM T63609 CB9O5T 137370896 IC50 = 8200 nM T44614 D09EGZ 2719 IC50 = 20 nM T44614 CH0CT9 300140 IC50 = 20800 nM T44614 C6B5KN 439487 IC50 = 68 nM T44614 CX06HK 701796 IC50 = 29600 nM T44614 C4X1BC 704553 IC50 = 22500 nM T44614 C47PBN 715039 IC50 = 38600 nM T44614 CU4M6G 766854 IC50 = 43900 nM T44614 C8YWA6 843629 IC50 = 28700 nM T44614 CZMJ46 855979 IC50 = 6670 nM T44614 CL2N7W 858292 IC50 = 6670 nM T44614 CH6BA5 867859 IC50 = 27300 nM T44614 CF6KH2 870542 IC50 = 13200 nM T44614 C6S3NJ 980900 IC50 = 1400 nM T44614 CSMN80 1018414 IC50 = 7500 nM T44614 C7P9LG 1069242 IC50 > 50000 nM T44614 CQJ2H6 1098384 IC50 = 40900 nM T44614 C0J2CX 1136480 IC50 = 6200 nM T44614 CZA7T4 1151414 IC50 = 12400 nM T44614 C3EX8R 1169419 IC50 = 6670 nM T44614 C5O3QY 1377557 IC50 = 2100 nM T44614 C7IOQ9 1377754 IC50 = 4600 nM T44614 C7KZ3E 1440076 IC50 = 6670 nM T44614 C2FKL0 1463717 IC50 = 6670 nM T44614 CY43VS 1463844 IC50 = 6670 nM T44614 CA3OK0 1734060 IC50 = 6500 nM T44614 C0O4QG 2246214 IC50 = 53400 nM T44614 C4D9LG 2739885 IC50 = 5400 nM T44614 CST02U 2740447 IC50 = 47800 nM T44614 CAO35D 2764792 IC50 = 15300 nM T44614 C5MG7B 2807600 IC50 = 10400 nM T44614 CFQZ06 2808735 IC50 = 14300 nM T44614 CJ5N7Q 2810657 IC50 = 19000 nM T44614 CF1G4U 2812460 IC50 = 2900 nM T44614 CF5VS7 2814162 IC50 = 52300 nM T44614 CHL5U2 2819033 IC50 = 13200 nM T44614 CD6LG1 2820117 IC50 = 3400 nM T44614 C3H5ET 3136444 IC50 = 6670 nM T44614 CW3KL5 3166734 IC50 = 6670 nM T44614 CQ9CD1 3188643 IC50 = 6670 nM T44614 C3SD5C 3192819 IC50 = 6670 nM T44614 CRL3B6 3570088 IC50 = 1600 nM T44614 CQ0AR8 3704739 IC50 = 46900 nM T44614 CY0UX3 5332358 IC50 = 2200 nM T44614 CD39LW 5480198 IC50 > 20000 nM T44614 CH06BX 5506952 IC50 = 5700 nM T44614 CDT70P 5839370 IC50 = 50000 nM T44614 CDBE15 5947235 IC50 > 20000 nM T44614 C8B7TO 5984369 IC50 > 20000 nM T44614 CTEO56 6373261 IC50 = 6200 nM T44614 CHO4P1 7224671 IC50 = 10000 nM T44614 C6ZHR7 9553596 IC50 = 26600 nM T44614 C8Q5TO 9584421 IC50 = 54300 nM T44614 CQZ75R 9667011 IC50 = 10800 nM T44614 C47KUQ 10471660 IC50 = 9200 nM T44614 CJ97UE 10705932 IC50 = 40000 nM T44614 CV63PX 10782475 IC50 = 10000 nM T44614 C5E8FN 10793407 IC50 = 7330 nM T44614 CY40NC 11065815 IC50 = 30000 nM T44614 COA2Y3 11172107 IC50 > 20000 nM T44614 C3DV9K 11176351 IC50 = 3800 nM T44614 CNM0X6 11199052 IC50 > 20000 nM T44614 CN0F8E 11199915 IC50 = 5000 nM T44614 CZ43RI 11293753 IC50 = 2500 nM T44614 C4V7LA 11315911 IC50 = 2600 nM T44614 CXWY85 11452912 IC50 = 2500 nM T44614 CR5WN3 11464039 IC50 = 2600 nM T44614 CUOZ49 11465492 IC50 = 1800 nM T44614 C5W8BG 11498009 IC50 = 8250 nM T44614 CGC36Z 11534339 IC50 = 15040 nM T44614 CE39KT 11556013 IC50 = 8790 nM T44614 C84JRM 11571002 Ki = 4000 nM T44614 C9MFO3 11591978 IC50 = 21540 nM T44614 CL8PI1 11592397 IC50 = 11190 nM T44614 CB0G5Y 11594647 IC50 = 620 nM T44614 C85WBA 11599792 Ki = 400 nM T44614 CJ4RW9 11612408 IC50 < 6600 nM T44614 CYAT21 11628282 IC50 = 16340 nM T44614 CVW4Z2 11628448 IC50 = 13510 nM T44614 CM0LH5 11650373 IC50 = 10290 nM T44614 CJ9FY4 11686106 IC50 = 19150 nM T44614 C5SZ9Q 11737693 IC50 > 20000 nM T44614 C71KNB 15984111 IC50 = 13700 nM T44614 CQ5F9T 16045426 IC50 = 0.6 nM T44614 CGTM78 24800873 Ki = 390 nM T44614 C1LOF2 24800874 Ki = 53 nM T44614 CMI4L3 24800875 Ki = 140 nM T44614 CAXQ09 24801230 Ki = 320 nM T44614 CT1A2Z 24801231 Ki = 600 nM T44614 C2O4WK 24801410 Ki = 370 nM T44614 C5NI0K 24801411 Ki = 110 nM T44614 CXB4D8 24825644 IC50 > 20000 nM T44614 CH8G0R 24825645 IC50 > 20000 nM T44614 CWY3S8 24825646 IC50 > 20000 nM T44614 CJ74RK 24825647 IC50 > 20000 nM T44614 CP67YX 24825648 IC50 > 20000 nM T44614 C73KLE 25209862 IC50 = 8.5 nM T44614 COB43C 25798545 IC50 = 34600 nM T44614 CLG09E 44391871 IC50 = 1800 nM T44614 C3LV8U 44391872 IC50 = 640 nM T44614 C5BW3L 44391882 IC50 = 375 nM T44614 C01MLD 44391883 IC50 = 2600 nM T44614 CZ63QT 44391902 IC50 = 14000 nM T44614 C5QR1V 44391906 IC50 = 470 nM T44614 C3T8YW 44391915 IC50 = 8400 nM T44614 CXBC18 44400441 IC50 = 12500 nM T44614 CFLY07 44400517 IC50 = 3400 nM T44614 CI6GH4 44408358 IC50 = 13800 nM T44614 CKC4P5 44411027 Ki = 43900 nM T44614 C2MDN7 44411237 Ki = 28300 nM T44614 C6H7ZT 44414312 IC50 = 23600 nM T44614 CV87SR 44414390 IC50 = 26500 nM T44614 CDAZ59 44414416 IC50 = 48400 nM T44614 CHMJ74 44414631 IC50 = 31400 nM T44614 C8IP6C 44444723 IC50 = 4416 nM T44614 C4JP1U 44444724 IC50 > 20000 nM T44614 C20FYI 44444725 IC50 = 12932 nM T44614 CJVK57 44444726 IC50 > 20000 nM T44614 C5I2XF 44457308 Ki = 120 nM T44614 CG76CX 44560637 IC50 = 10900 nM T44614 CT9ER7 44560638 IC50 = 19000 nM T44614 CFZB79 44572423 Ki = 17 nM T44614 C4HOQ6 46216666 IC50 > 100000 nM T44614 CNI30F 46216667 IC50 > 100000 nM T44614 C7GNS6 46230574 IC50 > 100000 nM T44614 C28PBV 46230575 IC50 > 100000 nM T44614 CW3EH5 46230576 IC50 > 100000 nM T44614 CV9YN2 46230577 IC50 > 100000 nM T44614 CFQ62C 46231266 IC50 > 100000 nM T44614 CS1AG6 46231303 IC50 > 100000 nM T44614 CJ9Q2P 46231304 IC50 > 100000 nM T44614 CPNJ84 46231305 IC50 > 100000 nM T44614 C0ZTC5 46231306 IC50 > 100000 nM T44614 CU59GB 46231307 IC50 > 19000 nM T44614 C9VB7F 46231308 IC50 > 100000 nM T44614 C0A6HL 46231345 IC50 > 100000 nM T44614 CB7N3J 46231346 IC50 > 100000 nM T44614 C8T7DK 46231347 IC50 > 100000 nM T44614 CYGB69 46231348 IC50 > 100000 nM T44614 C7VLI1 46231349 IC50 > 100000 nM T44614 C1HNB6 46838159 Ki = 8200 nM T44614 C2UOK6 46838161 Ki = 8900 nM T44614 C9LNK5 49798881 Ki = 1560 nM T44614 CE6Z7V 49798882 Ki > 100000 nM T44614 C5CY7U 49798883 Ki = 15100 nM T44614 C3B8FE 49798886 Ki = 3480 nM T44614 C8R6CQ 49798901 Ki > 100000 nM T44614 C7YZV2 49798902 Ki = 89000 nM T44614 CO7I0B 49798903 Ki = 14 nM T44614 CVT4U3 49798904 Ki = 2220 nM T44614 C3Y6OC 49798905 Ki = 460 nM T44614 C75LIT 59907274 IC50 > 50000 nM T44614 CW91LK 71463489 IC50 > 12500 nM T44614 CQ34FZ 71463490 IC50 = 39100 nM T44614 CIE54Z 71463491 IC50 > 33000 nM T44614 CR1WA0 71463492 IC50 > 33000 nM T44614 C05CUA 71463493 IC50 = 15300 nM T44614 CM1I0W 71463494 IC50 > 12500 nM T44614 CA87KS 71463495 IC50 > 33000 nM T44614 C7J2HR 76307998 IC50 = 890 nM T44614 C3G5OE 76307999 IC50 = 260 nM T44614 CQB6N0 76308000 IC50 = 170 nM T44614 CUVE40 76310777 IC50 > 50000 nM T44614 CWR65Z 76310778 IC50 > 50000 nM T44614 CE6N2S 76310779 IC50 = 80 nM T44614 CUE84S 76310780 IC50 > 50000 nM T44614 C70ZPY 76314405 IC50 > 50000 nM T44614 CNK1T8 76314406 IC50 = 3250 nM T44614 C2Q7AD 76314407 IC50 > 50000 nM T44614 CCAU01 76315163 IC50 = 150 nM T44614 CP3DL5 76315164 IC50 = 520 nM T44614 C8QYX9 76318812 IC50 = 840 nM T44614 C1PJB5 76318813 IC50 = 2280 nM T44614 CG8Q9N 76318814 IC50 = 390 nM T44614 CIG87S 76321694 IC50 > 50000 nM T44614 C43KMV 76321695 IC50 = 5520 nM T44614 CI4WD1 76321696 IC50 = 4420 nM T44614 CN91JU 76321697 IC50 > 50000 nM T44614 CAR0T5 76322470 IC50 = 210 nM T44614 CN3O4W 76322471 IC50 = 670 nM T44614 CNRS91 76325307 IC50 = 48130 nM T44614 CG2M0Z 76325308 IC50 = 33860 nM T44614 CLK1R8 76325309 IC50 = 29670 nM T44614 CO73BS 76326076 IC50 = 280 nM T44614 CSTH79 76326077 IC50 = 780 nM T44614 C58XRT 76328858 IC50 > 50000 nM T44614 C7UPX0 76328859 IC50 = 30080 nM T44614 CC2D7A 76328860 IC50 = 33640 nM T44614 CLY63W 76329664 IC50 = 290 nM T44614 CJ6P7X 76332528 IC50 > 50000 nM T44614 CNUO17 76332529 IC50 > 50000 nM T44614 CI41EG 76333338 IC50 = 840 nM T44614 CR6Q3G 76336143 IC50 > 50000 nM T44614 CS2L4D 76336144 IC50 = 1100 nM T44614 C95UVL 76336145 IC50 > 50000 nM T44614 C6A1TJ 102600382 Ki = 200 nM T44614 C0GOA7 102600383 Ki = 800 nM T44614 CMXE08 102600384 Ki = 1100 nM T44614 CJ1Q2F 118731975 Ki = 1800 nM T44614 CF62YN 118731976 Ki = 13600 nM T44614 CBO46Y 118731977 Ki = 6200 nM T44614 CT3L6R 118731978 Ki = 10600 nM T44614 C54PNI 118731979 Ki = 7000 nM T44614 C8IQ2N 118731980 Ki = 400 nM T44614 CIZA17 118731981 Ki = 400 nM T44614 CT5QJ0 118731982 Ki = 2530 nM T44614 CQ83OY 118731983 Ki = 3290 nM T44614 COH81Z 118731984 Ki = 7490 nM T44614 CEW7S2 118731985 Ki = 4600 nM T44614 C5Y4ZE 118731986 Ki = 1300 nM T44614 C5JDV0 118731987 Ki > 10000 nM T44614 CV9N4T 118731988 Ki > 10000 nM T44614 CH79SN 118731989 Ki > 100000 nM T44614 C5H7LC 118731990 Ki = 300 nM T44614 CU72OZ 118731991 Ki = 300 nM T44614 CWHE40 118731992 Ki = 800 nM T44614 C3KEF7 118731993 Ki = 600 nM T44614 CN5F2V 118732129 Ki = 8600 nM T44614 CHQ8O9 135400553 IC50 = 3900 nM T44614 CQDO50 135405855 IC50 = 7000 nM T44614 CT08UH 135406805 IC50 = 59900 nM T44614 CPL94A 135435989 IC50 = 4600 nM T44614 CGV4W2 135439445 IC50 = 32800 nM T44614 C3KNA4 135463520 IC50 = 3160 nM T44614 C0CM3I 135478389 IC50 = 63400 nM T44614 C72GEI 135492196 IC50 = 7500 nM T44614 CR07MW 135495603 IC50 = 31100 nM T44614 C7UKH0 135783341 IC50 = 11070 nM T44614 C49QTK 135783342 IC50 = 5850 nM T44614 CW24GK 135783343 IC50 = 3800 nM T44614 C19JQW 135783344 IC50 > 20000 nM T44614 C7RI8W 135783345 IC50 = 18220 nM T44614 CR0IU4 135783346 IC50 = 2250 nM T44614 C13VRH 135783347 IC50 > 20000 nM T44614 CN2TS3 135783348 IC50 = 2600 nM T44614 CO4ED1 135783349 IC50 = 720 nM T44614 CW21GB 135783350 IC50 = 630 nM T44614 CM67YW 135783351 IC50 > 20000 nM T44614 CB0W9I 135783352 IC50 > 20000 nM T44614 C4PMD2 135993358 IC50 > 20000 nM T44614 CGO97R 136029168 IC50 = 9400 nM T44614 CT39DN 137637025 IC50 > 50000 nM T44614 C39AXE 137637300 IC50 = 780 nM T44614 C5MF9X 137638638 IC50 = 1320 nM T44614 C25QTS 137639741 IC50 = 250 nM T44614 C6W7AO 137641179 IC50 > 50000 nM T44614 CQ8F4R 137643756 IC50 > 50000 nM T44614 C1AXD7 137647008 IC50 = 780 nM T44614 CZK74L 137647856 IC50 > 50000 nM T44614 CZBU13 137651934 IC50 = 3010 nM T44614 CS8U7B 137653242 IC50 > 50000 nM T44614 C5QVE7 137655537 IC50 = 110 nM T44614 CZA12J 137659286 IC50 > 50000 nM T44614 C2FGL6 137660813 IC50 = 9530 nM T44614 C6MI1F 137661465 IC50 = 9630 nM T44614 CR6PW7 145948246 IC50 = 7700 nM T44614 CHG1F4 145948247 IC50 = 3710 nM T44614 C3GA9W 145948249 IC50 = 10500 nM T44614 C0SU5G 145948250 IC50 > 50000 nM T44614 CK8GV9 145948253 IC50 = 11500 nM T44614 CDX4E1 145948254 IC50 = 3400 nM T44614 CRLB34 145948256 IC50 = 2500 nM T44614 CVW6F9 145948259 IC50 = 5.25 nM T44614 C7W6NP 145948265 IC50 = 12 nM T44614 CMX0N5 145948268 IC50 = 9.59 nM T44614 CDF1L7 145948270 IC50 = 6.86 nM T44614 CT7HX4 145948276 IC50 = 6.78 nM T44614 C4WLY7 145948278 IC50 = 2.81 nM T44614 CFQ25D 145967499 IC50 > 5000 nM T44614 CU0VZ4 145967573 IC50 = 2.2 nM T44614 CIVB10 145967715 IC50 = 57 nM T44614 C5Q8GV 145967809 IC50 = 14300 nM T44614 CLI6T0 145967952 IC50 = 178 nM T44614 CQT02S 145968345 IC50 = 8.2 nM T44614 CC4AG7 145968405 IC50 > 5000 nM T44614 C70IDL 145968427 IC50 = 10400 nM T44614 CDC09E 145968500 IC50 > 100000 nM T44614 C06DWX 145968519 IC50 = 20900 nM T44614 CZ3EQ6 145968606 IC50 = 2.4 nM T44614 CDS31M 145968622 IC50 = 27 nM T44614 CQ9U4N 145968625 IC50 > 5000 nM T44614 C7CEA8 145968774 IC50 = 25.9 nM T44614 CKN52D 145968813 IC50 = 1.2 nM T44614 C5X0OJ 145968845 IC50 = 26900 nM T44614 CT5GM7 145968865 IC50 = 3 nM T44614 C0F4GN 145968902 IC50 > 100000 nM T44614 C2WH6O 145969099 IC50 = 3300 nM T44614 CA40YU 145969275 IC50 = 667 nM T44614 CIO4A9 145969330 IC50 = 26700 nM T44614 C4H0GF 145969424 IC50 = 34200 nM T44614 CB0Y7Z 145969438 IC50 > 5000 nM T44614 C2WCK0 145969450 IC50 = 1585 nM T44614 CN4OR1 145969487 IC50 > 100000 nM T44614 C5F2PY 145969506 IC50 = 17500 nM T44614 CYZ10E 145969765 IC50 = 8.6 nM T44614 CL7KO9 145969878 IC50 = 137 nM T44614 CULQ78 145969983 IC50 = 6.3 nM T44614 C3NAS7 145970030 IC50 > 5000 nM T44614 CW16PV 145970433 IC50 = 55.4 nM T44614 CEV41D 145970469 IC50 = 18600 nM T44614 CK9BE1 145970625 IC50 = 4200 nM T44614 CR83BK 145970650 IC50 = 2.7 nM T44614 CS08XI 145970918 IC50 > 5000 nM T44614 C9XKW2 145970931 IC50 = 192 nM T44614 C5CYV4 145971156 IC50 = 19700 nM T44614 C5XQ6R 145971181 IC50 > 100000 nM T44614 CE3GW7 145981911 Ki = 1260 nM T44614 C6OKB9 145987263 IC50 > 5000 nM T44614 CEYU65 145987330 Ki = 28600 nM T44614 COZ6P5 145987960 IC50 = 230 nM T44614 C7ZCW3 145988622 IC50 > 5000 nM T44614 C9OAK6 145989037 IC50 = 8 nM T44614 C87GKT 145989707 IC50 = 23.1 nM T44614 CH7WO9 145994261 Ki = 450 nM T44614 CIGE48 155510826 IC50 = 29 nM T44614 C1M3XR 155512606 IC50 = 235 nM T44614 C1XP0B 155513744 IC50 = 33 nM T44614 CO6JQ0 155515904 IC50 = 84 nM T44614 C02OMN 155516116 IC50 = 57 nM T44614 C32YQR 155520783 IC50 = 6670 nM T44614 C8J7WI 155525675 IC50 = 270 nM T44614 CW1C9V 155532002 IC50 = 31 nM T44614 CSN35Y 155535964 IC50 = 59 nM T44614 CC5UP3 155536311 IC50 = 3097 nM T44614 CYZD26 155537774 IC50 = 464 nM T44614 C8GK9E 155540750 IC50 = 169 nM T44614 C17BLD 155544667 IC50 = 156 nM T44614 C1IKN8 155556814 IC50 = 455 nM T44614 CZAE90 155556984 IC50 > 50000 nM T44614 C25OHZ 155559205 IC50 = 60 nM T44614 CWU5L7 155559556 IC50 > 50000 nM T44614 CDH54L 155569478 IC50 = 3523 nM T44614 C5ZSA0 118722665 IC50 = 6000 nM T44614 CO5UD0 118722667 IC50 > 50000 nM T44614 CX8EU0 118722669 IC50 > 50000 nM T44614 C3TL8E 118722671 IC50 = 24.8 nM T44614 C5FB8V 118722672 IC50 = 9.52 nM T44614 CHN97M 13339465 IC50 > 50000 nM T44614 C2PU5B 13339466 IC50 > 50000 nM T44614 C61UIJ 13339468 IC50 > 50000 nM T44614 C63ZMF 4388929 IC50 = 4400 nM T44614 CWKQ68 51355958 IC50 > 50000 nM T44614 CG36ZN 51355959 IC50 > 50000 nM T44614 CSR1J3 728912 IC50 > 50000 nM T44614 D01BQI 25798544 IC50 = 21900 nM T44614 D08KCA 72429 IC50 = 87 nM T44614 D09FGQ 123985 IC50 = 15 nM T44614 D0G2DQ 4669250 IC50 = 42600 nM T44614 D0L9VP 5287864 IC50 = 2 nM T44614 D0O5TA 2175573 IC50 = 31200 nM T44614 D0TZ5V 690109 IC50 = 38800 nM T48812 D02DGU 444795 IC50 = 0.15 nM T48812 D0D7CH 118622692 IC50 >= 30000 nM T48812 C25CAT 122184111 EC50 = 1300 nM T48812 CVS15Y 122184115 EC50 = 1700 nM T48812 C6R8ES 72721387 EC50 = 1930 nM T48812 C2LMW1 18565134 EC50 = 4100 nM T48812 C0QKH8 18565138 EC50 = 5400 nM T48812 CGS1R9 18565141 EC50 = 3400 nM T48812 C4RYO8 19760309 IC50 > 10000 nM T48812 C38JEL 20704150 EC50 = 4000 nM T48812 C1FJU8 21824365 IC50 = 13400 nM T48812 CF1S8P 25132150 IC50 > 20000 nM T48812 CNG1Z5 25132504 IC50 = 10100 nM T48812 CB56QH 25132505 IC50 > 20000 nM T48812 CS1EJ7 25234324 EC50 = 5000 nM T48812 CO1NQ0 41145803 IC50 = 1995.26 nM T48812 C9ZWM8 46866594 IC50 = 6500 nM T48812 CMR49F 46885348 IC50 > 20000 nM T48812 C18JYQ 46885349 IC50 = 8800 nM T48812 C4TLX3 46885390 IC50 = 17100 nM T48812 CSP3D8 46885467 IC50 = 7900 nM T48812 C8WM2R 46885468 IC50 = 17000 nM T48812 CP3O2L 46885469 IC50 > 20000 nM T48812 CG6JE7 46885508 IC50 = 12800 nM T48812 CX2U0L 46886033 IC50 > 20000 nM T48812 C6J5RT 46886034 IC50 = 5400 nM T48812 C2P5HX 54582225 IC50 = 10900 nM T48812 CQ02IF 54582227 IC50 > 10000 nM T48812 CS9O7F 54582228 IC50 = 7700 nM T48812 CPF9X2 54587076 IC50 = 7500 nM T48812 CFO23H 56837193 IC50 = 64 nM T48812 CJ0I1V 71082496 IC50 = 11300 nM T48812 CXK08C 71612420 EC50 = 2700 nM T48812 C1DR8E 71622396 EC50 = 2500 nM T48812 CWH6T3 72548703 IC50 = 164 nM T48812 CIV80W 72548704 IC50 = 326 nM T48812 CZ0P6M 72548955 IC50 = 230 nM T48812 CC8YU6 72720884 EC50 = 1100 nM T48812 CMZ85K 72722807 EC50 = 5000 nM T48812 C2BQO3 72722945 EC50 = 6000 nM T48812 C6UWO5 74762670 EC50 = 3800 nM T48812 CJXG25 76284182 EC50 > 10000 nM T48812 C5PT4U 76314451 IC50 > 10000 nM T48812 CMW6O1 77620538 EC50 = 2200 nM T48812 C7ZMD9 78319220 IC50 = 4900 nM T48812 C4SA8H 86302482 EC50 > 10000 nM T48812 CBI06J 86346645 EC50 > 10000 nM T48812 C5VCM4 86690644 EC50 > 10000 nM T48812 CGFW70 86690646 EC50 > 10000 nM T48812 CNL0R1 87074581 IC50 = 59 nM T48812 CXO3F6 87085264 IC50 = 610 nM T48812 C5DW8X 87085361 IC50 = 240 nM T48812 C5MOV2 89659415 EC50 = 1200 nM T48812 CLW3O5 89665055 EC50 = 3700 nM T48812 C7E5RV 90200534 EC50 > 10000 nM T48812 CBCE70 90465832 IC50 > 30000 nM T48812 CEB82Q 90646513 IC50 > 30000 nM T48812 C0Z4BC 90646903 IC50 > 30000 nM T48812 C9FQ2N 90656122 IC50 = 11800 nM T48812 CF4M9V 90656123 IC50 = 9700 nM T48812 C5E6UV 90656124 IC50 = 8200 nM T48812 CS43BG 90656125 IC50 = 7100 nM T48812 C9TI2B 90656126 IC50 = 5600 nM T48812 C35ICO 90656127 IC50 = 5500 nM T48812 CI92WR 91664317 EC50 > 10000 nM T48812 C4S9EM 117964962 EC50 > 10000 nM T48812 CS4GJ9 117964973 EC50 > 10000 nM T48812 CDXK37 117964975 EC50 > 10000 nM T48812 CN6RT8 117964978 EC50 > 10000 nM T48812 C96BSK 117964998 EC50 > 10000 nM T48812 CKT50F 118185722 IC50 = 154 nM T48812 CG7FY8 118185723 IC50 = 425 nM T48812 CKCO28 118185739 IC50 = 163 nM T48812 CI3L8V 118185743 IC50 = 83 nM T48812 C3Z8WU 118185750 IC50 = 115 nM T48812 CML8Q4 118186054 IC50 = 176 nM T48812 CDF8G3 118188696 IC50 = 119 nM T48812 C79IOD 118207841 EC50 > 40000 nM T48812 C2FLM1 118207907 EC50 > 40000 nM T48812 CXW5M0 118207954 EC50 > 40000 nM T48812 C9UK5A 118207966 EC50 > 40000 nM T48812 C0PWH6 118207991 EC50 > 40000 nM T48812 C2U3TJ 118208018 EC50 > 40000 nM T48812 CZ2C3U 118208048 EC50 > 40000 nM T48812 C8N2PF 118208184 EC50 > 40000 nM T48812 C1ZRN9 118217594 EC50 > 40000 nM T48812 CAUT58 118217595 EC50 > 40000 nM T48812 CCK3J9 118217851 EC50 > 40000 nM T48812 CO5I3V 118217852 EC50 > 40000 nM T48812 CD5TJ3 118217853 EC50 > 40000 nM T48812 C6HSC3 118217854 EC50 > 40000 nM T48812 CEKH57 118217858 EC50 > 40000 nM T48812 C1CTB6 118217859 EC50 > 40000 nM T48812 C7U0XR 118217863 EC50 > 40000 nM T48812 CDP0H5 118217865 EC50 > 40000 nM T48812 C82YDU 118217866 EC50 > 40000 nM T48812 CQ60HK 118217867 EC50 > 40000 nM T48812 C9N7VY 118217868 EC50 > 40000 nM T48812 C6LC7H 118217869 EC50 > 40000 nM T48812 CV9G4S 118217870 EC50 > 40000 nM T48812 C8PR3G 118217871 EC50 > 40000 nM T48812 CZ3FX6 118217874 EC50 > 40000 nM T48812 CT0DV4 118217911 EC50 > 40000 nM T48812 C1QPW5 118217915 EC50 > 40000 nM T48812 C3YTM2 118217920 EC50 > 40000 nM T48812 CU0T7K 118217922 EC50 > 40000 nM T48812 C0ETA2 118217925 EC50 > 40000 nM T48812 C6X4IN 118217935 EC50 > 40000 nM T48812 CD01CA 118526849 EC50 > 8000 nM T48812 CBZ75K 118724654 EC50 > 3100 nM T48812 CB0AH7 118865631 IC50 > 30000 nM T48812 C27MYR 118865641 IC50 > 30000 nM T48812 C6TBD2 121345502 EC50 > 20000 nM T48812 CO6HF9 122180196 IC50 = 6700 nM T48812 CEW72J 122180199 IC50 = 7000 nM T48812 C5L1AS 122184114 EC50 = 1100 nM T48812 CL7EY2 122184139 EC50 = 2300 nM T48812 CE87BY 122184140 EC50 = 800 nM T48812 CRY8N5 122190169 EC50 = 7900 nM T48812 C0WAM1 122379290 EC50 = 5400 nM T48812 C4F9ZK 122669103 IC50 > 10000 nM T48812 CZH39M 122669106 IC50 > 10000 nM T48812 C0T8FO 122669173 IC50 > 10000 nM T48812 CD6X5P 122669265 EC50 > 10000 nM T48812 C0S7UB 122678562 IC50 > 10000 nM T48812 CY8S1P 122678563 IC50 > 10000 nM T48812 C0MUW2 122678576 IC50 > 10000 nM T48812 C2SQ9M 122678748 IC50 > 10000 nM T48812 CH1J6K 122678779 IC50 > 10000 nM T48812 CD9HN3 122678983 IC50 > 10000 nM T48812 CF39TE 122679031 IC50 > 10000 nM T48812 C0XWI7 127029952 IC50 = 60000 nM T48812 CB3HG0 134817247 IC50 > 10000 nM T48812 CK3X1N 137796283 IC50 > 10000 nM T48812 CJ2R7W 141493565 EC50 > 10000 nM T48812 C7XT6D 141493567 EC50 > 10000 nM T48812 CC2BH9 145232219 IC50 > 10000 nM T48812 CW3Y0H 145949340 IC50 > 20000 nM T48812 CPK5U1 145951022 IC50 > 20000 nM T48812 CKT24R 145951943 IC50 > 20000 nM T48812 CR70ZO 145957041 IC50 > 10000 nM T48812 C60CMX 145958026 IC50 > 10000 nM T48812 CL2HT7 145959111 IC50 > 10000 nM T48812 CIMW18 145961622 IC50 = 13 nM T48812 CJ7RU8 145961892 IC50 = 184 nM T48812 C56QRW 145962236 IC50 = 940 nM T48812 CWRU80 145962336 IC50 = 53 nM T48812 CEU4V3 145962457 IC50 = 16 nM T48812 CN7Z3Q 145963286 IC50 = 490 nM T48812 C01QZJ 145963443 IC50 = 3.4 nM T48812 C4H9UY 145966156 EC50 > 2000 nM T48812 CO02AH 145967656 IC50 = 63 nM T48812 C4JZ8T 145967902 IC50 = 120 nM T48812 CTAP43 145968298 IC50 = 290 nM T48812 CKT3A4 145968585 IC50 = 110 nM T48812 CBQ91G 145968987 IC50 = 160 nM T48812 C0GX6M 145969292 IC50 = 310 nM T48812 CUV3R6 145969329 IC50 = 140 nM T48812 C76RKW 145969356 IC50 = 130 nM T48812 C6CFJ8 145969713 IC50 = 290 nM T48812 CX7GL1 145970040 IC50 = 410 nM T48812 C7VJM9 145970264 IC50 = 1400 nM T48812 CFK76Y 145970594 IC50 = 90 nM T48812 CXE10U 145970665 IC50 = 410 nM T48812 CGR9U4 145970687 IC50 = 160 nM T48812 CPJI78 145971170 IC50 = 370 nM T48812 CD37PO 145979241 IC50 = 230 nM T48812 CB70AE 145980094 IC50 > 10000 nM T48812 CXW29A 145982397 IC50 = 130 nM T48812 C5VBU6 145982695 IC50 = 200 nM T48812 C1JUC8 145982712 IC50 > 30000 nM T48812 CUN03M 145982910 IC50 = 360 nM T48812 C89ZMA 145985638 IC50 = 40 nM T48812 CRTG03 145987785 IC50 > 10000 nM T48812 CAU45I 145987980 IC50 < 10 nM T48812 C8C5KF 145988118 IC50 = 90 nM T48812 CM0G9W 145988515 IC50 = 76 nM T48812 C4ESM8 145988957 IC50 = 15 nM T48812 CDI01N 145989245 IC50 = 220 nM T48812 C5KG8D 145989415 IC50 = 240 nM T48812 CWSP97 145989563 IC50 = 180 nM T48812 CVHY07 145989633 IC50 = 980 nM T48812 C7HGR2 145989697 IC50 = 26 nM T48812 CG02OC 145990362 IC50 = 330 nM T48812 CCYQ80 145990612 IC50 = 380 nM T48812 C4W7IA 145991126 IC50 = 90 nM T48812 C50IES 145991139 IC50 = 2600 nM T48812 CC4DV9 145991246 IC50 = 180 nM T48812 C5LXE1 145991424 IC50 = 570 nM T48812 CY58DQ 145991674 IC50 = 34 nM T48812 CVCR42 145991755 IC50 = 800 nM T48812 CP0FK5 145991857 IC50 = 94 nM T48812 C0EB5D 145992591 IC50 = 87 nM T48812 C3Q0ZN 145993067 IC50 = 230 nM T48812 C67AUF 145993523 IC50 = 470 nM T48812 CKL05T 145994203 IC50 = 2400 nM T48812 CC89OI 148034311 IC50 > 10000 nM T48812 CUFS62 155510496 EC50 = 6800 nM T48812 CE6V8Z 155511797 IC50 > 10000 nM T48812 CU5Z8T 155522788 IC50 > 10000 nM T48812 C1DT9M 155525669 IC50 > 10000 nM T48812 CXS9T8 155526989 IC50 > 10000 nM T48812 CO9N5H 155530678 IC50 > 10000 nM T48812 CIUA10 155537856 IC50 > 10000 nM T48812 CLO98T 155539150 EC50 > 40000 nM T48812 COP7X8 155539171 IC50 > 10000 nM T48812 C0V6EY 155543172 IC50 > 10000 nM T48812 CX7L0S 155544387 IC50 > 10000 nM T48812 CSK20E 155544524 IC50 > 10000 nM T48812 CBK1E5 155556708 IC50 > 10000 nM T48812 C3FI7U 155560819 IC50 > 10000 nM T48812 CA91EM 155564933 IC50 > 10000 nM T48812 CPF42S 155565257 IC50 > 10000 nM T48812 C6KMU5 122184108 EC50 = 900 nM T48812 CV5CO0 122184112 EC50 = 1000 nM T48812 C63QAO 122184113 EC50 = 800 nM T48812 CT3WD4 122184116 EC50 = 600 nM T48812 CBHT23 122184117 EC50 = 1500 nM T48812 CH1EJ7 122184118 EC50 = 6200 nM T48812 C13QFC 122184133 EC50 = 1300 nM T48812 CO82BL 122184137 EC50 = 1800 nM T48812 CPM90L 122184138 EC50 = 1300 nM T48812 D0B5FC 447912 EC50 = 6000 nM T70234 D03LWG 53235510 IC50 > 10000 nM T70234 D07EHV 44814409 IC50 > 10000 nM T70234 D07HPJ 11476171 IC50 > 10000 nM T70234 D0E3TC 44259 IC50 = 12.5 nM T70234 D0T3ME 156422 IC50 = 70 nM T70234 CACS26 11561968 Ki > 10000 nM T70234 CU0E8O 11690457 Ki > 10000 nM T70234 C2W9OA 53324451 IC50 > 10000 nM T70234 C8NA4L 53384644 IC50 > 30000 nM T70234 C79LYD 53497554 IC50 = 4500 nM T70234 C87YOZ 56929808 IC50 = 74 nM T70234 C1Y7NU 56969069 IC50 = 2000 nM T70234 CTP19M 57345507 IC50 = 8100 nM T70234 C1MR8Q 60097495 IC50 > 10000 nM T70234 C1HSE0 67035086 IC50 = 9 nM T70234 CWI6K5 67035106 IC50 > 10000 nM T70234 C38RGB 67035556 IC50 = 4700 nM T70234 CV63UL 67240318 IC50 > 10000 nM T70234 C8I7GC 68293638 IC50 > 10000 nM T70234 CD56XK 68293660 IC50 > 10000 nM T70234 CYT52O 117072322 IC50 = 27 nM T70234 C9WGB8 127035904 IC50 = 3800 nM T70234 CTJ48K 135524085 IC50 = 5600 nM T70234 CUT1W7 135524168 IC50 > 10000 nM T70234 CSC5F6 155510719 IC50 = 54 nM T70234 C6A4RI 155511767 IC50 = 83 nM T70234 C2MD1Q 155513187 IC50 > 10000 nM T70234 CZ23CJ 155514081 IC50 = 25 nM T70234 C0E9FN 155516258 IC50 = 450 nM T70234 CSAO42 155519970 IC50 = 38 nM T70234 C4ET7C 155521014 IC50 = 50 nM T70234 CWR5O4 155526603 IC50 = 34 nM T70234 CFL56J 155528862 IC50 = 12 nM T70234 CHG7Z6 155531027 IC50 = 22 nM T70234 C0YUX8 155531038 IC50 = 17 nM T70234 C57LDI 155532993 IC50 > 10000 nM T70234 C20IUL 155537078 IC50 = 230 nM T70234 CQ23RB 155538387 IC50 = 1200 nM T70234 CN8UA9 155540659 IC50 = 41 nM T70234 CH8D4C 155541987 IC50 = 260 nM T70234 CYVN19 155542999 IC50 = 480 nM T70234 CVOG25 155546122 IC50 = 12 nM T70234 C2X9QO 155549598 IC50 = 40 nM T70234 C57HPY 155551696 IC50 = 290 nM T70234 C41CZQ 155568470 IC50 = 920 nM T70234 D05FXD 44478401 IC50 = 3.3 nM T70234 D06HVH 54613583 IC50 > 10000 nM T70234 D0X8BU 71718651 IC50 = 2700 nM T74500 D00PEH 135449332 IC50 = 1584893.19 nM T74500 D00STL 644241 IC50 = 3162277.66 nM T74500 D01AXB 60835 IC50 = 100000 nM T74500 D03IGH 213039 IC50 = 100000 nM T74500 D09MWJ 2092 IC50 = 1000000 nM T74500 D0B3UJ 115237 IC50 = 63095.73 nM T74500 D0BP9C 193962 IC50 = 3162277.66 nM T74500 D0BZ7W 443879 IC50 = 12589.25 nM T74500 D0C9SY 135400189 IC50 = 79432.82 nM T74500 D0E6XR 3062316 IC50 = 316227.77 nM T74500 D0I1FQ 54671008 IC50 = 5011872.34 nM T74500 D0K3QS 6442177 IC50 = 10000000 nM T74500 D0L4YD 154059 IC50 = 50118.72 nM T74500 D0O3FG 125017 IC50 = 5011872.34 nM T74500 D0Q5UQ 214348 IC50 = 50118.72 nM T74500 D0R0MW 5329102 IC50 = 50118.72 nM T74500 D0U0VU 5312125 IC50 = 316227.77 nM T74500 D0U2JP 4369359 IC50 = 100000000 nM T74500 D0X5ZI 6918493 IC50 = 251188.64 nM T74500 D0Y5AM 444031 IC50 = 12589.25 nM T74500 D0Z1UA 71301 IC50 = 50118.72 nM T74500 D0Z7ZM 135398744 IC50 = 501187.23 nM T74500 D02AIN 122678117 IC50 > 33000 nM T74500 CP8F7B 64143 IC50 = 5011872.34 nM T74500 CU7B8I 11525190 IC50 = 2300 nM T74500 CD34SB 15982534 IC50 > 100000 nM T74500 C8T4JF 16722295 IC50 = 8300 nM T74500 C91QFN 25019282 IC50 = 3870 nM T74500 CL41FE 46206000 IC50 > 100000 nM T74500 CA07TC 71517197 IC50 > 33000 nM T74500 CHD26A 121596332 IC50 > 33300 nM T74500 C1YK2E 122678192 IC50 > 33000 nM T74500 C4Z5MQ 131839619 IC50 > 30000 nM T74500 C8RFM3 145973261 IC50 > 33000 nM T74500 CG8I5F 155538033 IC50 = 11000 nM T74500 CKZT21 155559364 IC50 > 33000 nM T74500 D08HPL 6604863 IC50 = 1400 nM T46515 D03JSJ 446596 IC50 = 0.8 nM T46515 D0N1BC 9939559 IC50 = 0.00295 ug.mL-1 T46515 CP2U0R 9872941 IC50 = 0.0579 ug.mL-1 T46515 C4UX0T 9983945 IC50 = 30 nM T46515 C9X8NS 10005608 IC50 = 100 nM T46515 CH8M5T 10088604 IC50 = 4500 nM T46515 CP1ER7 10095725 IC50 = 98 nM T46515 CYW76I 10258978 IC50 = 0.211 ug.mL-1 T46515 CN9S6Y 10326551 IC50 = 0.4974 ug.mL-1 T46515 CWL8B6 10368969 IC50 = 300 nM T46515 CT9R2F 10415433 IC50 = 300 nM T46515 CU9WB0 10459578 IC50 = 100 nM T46515 C3OE6D 10865248 IC50 > 1 ug.mL-1 T46515 C2A7PI 11354737 IC50 > 1 ug.mL-1 T46515 CQ2W6P 11706052 IC50 > 1 ug.mL-1 T46515 C1TCX5 11848157 IC50 = 0.5645 ug.mL-1 T46515 C2S6XB 15514916 IC50 > 1 ug.mL-1 T46515 CWR60K 15514918 IC50 > 1 ug.mL-1 T46515 CTI4D2 24863020 IC50 = 0.0116 ug.mL-1 T46515 C01BXP 44327258 IC50 = 3000 nM T46515 CL7I2A 44327531 IC50 > 20000 nM T46515 CK1L4W 44341516 IC50 > 1 ug.mL-1 T46515 C7BA5J 44341566 IC50 = 0.0946 ug.mL-1 T46515 CJA5B8 44341898 IC50 = 0.374 ug.mL-1 T46515 C20TUP 44349029 IC50 = 45 nM T46515 C2JP3R 44349068 IC50 = 15 nM T46515 CB48XY 44349091 IC50 = 100 nM T46515 CM1R0V 44349092 IC50 > 100000 nM T46515 CC5RD8 44349103 IC50 = 100 nM T46515 CTYC72 44349104 IC50 = 100000 nM T46515 C9PN3I 44349131 IC50 = 20 nM T46515 C5KAZ8 44349132 IC50 = 1020 nM T46515 C0L8TO 44349189 IC50 > 100000 nM T46515 C3HK0S 44349205 IC50 = 15000 nM T46515 C5XM8K 44349437 IC50 = 120 nM T46515 CAC42O 44384563 IC50 = 181000 nM T46515 C37LTE 44384617 IC50 > 128000 nM T46515 C5BDC6 44384623 IC50 > 128000 nM T46515 C9C6NS 44384778 IC50 > 128000 nM T46515 CU9D5C 44384821 IC50 = 84000 nM T46515 CJHP70 44384945 IC50 > 128000 nM T46515 CV56PJ 44385054 IC50 = 228000 nM T46515 CHKJ16 44385230 IC50 = 57600 nM T46515 CCU8E6 44385306 IC50 = 45000 nM T46515 C7XY4F 44385414 IC50 > 128000 nM T46515 C7I1FJ 44385788 IC50 = 12800 nM T46515 CL59NH 44385851 IC50 = 106000 nM T46515 C5PSI9 44385912 IC50 = 21000 nM T46515 CYNV10 44385960 IC50 = 183000 nM T46515 CPY1K7 44386065 IC50 = 63600 nM T46515 C2IO8N 44386110 IC50 = 56500 nM T46515 CRB75J 44386149 IC50 > 128000 nM T46515 CJD0G1 44386211 IC50 = 64400 nM T46515 CT9J1G 44561404 IC50 > 1 ug.mL-1 T46515 CGM56A 44561405 IC50 = 0.2928 ug.mL-1 T46515 C2JOZ0 44561406 IC50 = 0.3783 ug.mL-1 T46515 CB5WR3 44561407 IC50 = 0.0583 ug.mL-1 T46515 CJKN52 44561408 IC50 = 0.0144 ug.mL-1 T46515 C9RNS3 44561409 IC50 = 0.0229 ug.mL-1 T46515 CPG0K4 44561410 IC50 = 0.5603 ug.mL-1 T46515 CS68WJ 44561411 IC50 > 1 ug.mL-1 T46515 CC8H3F 44561412 IC50 > 1 ug.mL-1 T46515 C2WA5Z 44561455 IC50 > 1 ug.mL-1 T46515 CI73OR 46874908 IC50 = 14 nM T46515 CEV78O 46874912 IC50 = 5500 nM T46515 CK94BH 46874919 IC50 = 12800 nM T46515 CVO1Q9 46874920 IC50 = 22200 nM T46515 CN2A7J 46874932 IC50 = 39 nM T46515 CPE89V 46874938 IC50 = 132000 nM T46515 CDL08S 46874966 IC50 = 1100 nM T46515 CD8JX1 135995964 IC50 = 50000 nM T46515 CQ45PG 135995968 IC50 = 79000 nM T46515 CP8EX0 135995970 IC50 = 38600 nM T92460 D0B3HD 2519 Ki = 10200 nM T92460 D04RKW 68374 Ki = 5550 nM T92460 D0M3IN 1188 Ki = 1960 nM T92460 CC7AH8 9679 Ki = 4440 nM T92460 CZJ8U9 30976 Ki = 1880 nM T92460 CX7JI2 128950 IC50 = 5000 nM T92460 C54RKT 9992468 Ki = 227000 nM T92460 CK9W0Z 16126716 Ki = 20100 nM T92460 CUY45C 44419607 Ki = 53600 nM T92460 C4OF1W 53323416 Ki = 16700 nM T92460 CK25WM 135432176 Ki = 3440 nM T92460 D0D3CS 1175 Ki = 4340 nM T46526 CVUJ20 89049 IC50 = 150 nM T46526 CF82PW 101798 IC50 = 1900 nM T46526 CR4H0V 46838220 IC50 = 1350 nM T46526 C2QE4F 46893411 IC50 = 144 nM T46526 C8CAV3 49855777 IC50 = 210 nM T46526 C83NMQ 49855778 IC50 = 253 nM T46526 CV06CI 49856159 IC50 = 9000 nM T46526 CUF74P 49856160 IC50 = 22 nM T46526 C2M0AH 49856161 IC50 = 16 nM T46526 CBC12X 49856162 IC50 = 15.3 nM T46526 CKU17I 49856163 IC50 = 45000 nM T46526 C7DTC4 49856165 IC50 = 10000 nM T46526 CA0I3U 49856349 IC50 = 27.6 nM T46526 CYV2I1 49856351 IC50 = 23.9 nM T46526 CBXZ63 49856356 IC50 = 31000 nM T46526 C1BIN7 49856544 IC50 = 38.7 nM T46526 CTY5J7 49856546 IC50 = 29.2 nM T46526 C5L9PW 56946890 IC50 = 70 nM T46526 C18ZUS 57390342 IC50 = 778 nM T46526 C79JHU 57392106 IC50 = 397 nM T46526 CXL76W 57392120 IC50 = 196 nM T46526 C8CUR9 57392121 IC50 = 565 nM T46526 CQF2J0 57393888 IC50 = 216 nM T46526 C95GDQ 57393889 IC50 = 333 nM T46526 CZE16F 57393890 IC50 = 327 nM T46526 CW3KE0 57395614 IC50 = 348 nM T46526 CB8RO9 57395615 IC50 = 153 nM T46526 CM0Z4G 57395644 IC50 = 296 nM T46526 C48ZAY 57397423 IC50 = 161 nM T46526 CS10UO 57397424 IC50 = 229 nM T46526 CR8DC9 57397425 IC50 = 250 nM T46526 CX7N6A 57397426 IC50 = 248 nM T46526 CBMA79 57397427 IC50 = 560 nM T46526 C15ACH 57397428 IC50 = 194 nM T46526 C5OHY0 57397454 IC50 = 207 nM T46526 C8DI0U 57397456 IC50 = 667 nM T46526 CCU2S1 57399085 IC50 = 511 nM T46526 CH93XY 57399104 IC50 = 639 nM T46526 C75GKL 57399129 IC50 = 420 nM T46526 CI1GH9 57400846 IC50 = 112 nM T46526 CTV62H 57402584 IC50 = 452 nM T46526 C8UVM4 57402608 IC50 = 331 nM T46526 C2VHA5 57402640 IC50 = 493 nM T46526 C2BK9D 57402641 IC50 = 169 nM T46526 C1DI3L 57402643 IC50 = 135 nM T46526 C9XMK1 57413864 IC50 = 150 nM T46526 CQ7H4I 76310828 IC50 = 58 nM T46526 C4KA5F 76310829 IC50 = 746 nM T46526 CK7GZ9 76310830 IC50 = 105 nM T46526 CPNL61 76314448 IC50 = 978 nM T46526 CWG83I 76318036 IC50 = 472 nM T46526 C7U3FD 76318038 IC50 = 804 nM T46526 C6GCM4 76321751 IC50 = 607 nM T46526 CGE2N3 76321752 IC50 = 144 nM T46526 C06FQB 76325364 IC50 = 763 nM T46526 CNL49F 76325365 IC50 = 450 nM T46526 CUS61H 76325366 IC50 = 593 nM T46526 CCY93X 76325367 IC50 = 875 nM T46526 CK6RA9 76332597 IC50 = 536 nM T46526 CBQ51T 86344039 IC50 = 130 nM T46526 C3PIQ0 101884902 IC50 = 346 nM T46526 CO4LY0 101884903 IC50 = 232 nM T46526 CRY0J4 122182804 IC50 = 208 nM T46526 CX9KR6 122182805 IC50 = 158 nM T46526 CCK60P 122182806 IC50 = 212 nM T46526 CVA62Z 130408860 IC50 = 40 nM T46526 C9GZ5H 130408883 IC50 = 38000 nM T46526 C84UAQ 130408935 IC50 = 40 nM T46526 CWO46P 130408951 IC50 = 11000 nM T46526 CTD03O 130408992 IC50 = 30 nM T46526 C8QV3R 130409041 IC50 = 900 nM T46526 CY97ER 130409062 IC50 = 600 nM T46526 C6RK5S 130409082 IC50 = 80 nM T46526 CE5C6Q 130455396 IC50 = 140 nM T46526 C40EIS 132281908 IC50 = 640 nM T46526 C6SXY2 134132865 IC50 = 250 nM T46526 CRY80S 134137026 IC50 = 340 nM T46526 C6Z8AC 139030264 IC50 = 280 nM T46526 C2AHJ8 139030265 IC50 = 2200 nM T46526 CGL3K2 139030266 IC50 = 34000 nM T46526 CZCV59 142590090 IC50 = 310 nM T46526 C2S3FH 142590102 IC50 = 510 nM T46526 C9TCY4 142590116 IC50 = 3500000 nM T46526 C5TX0P 142590121 IC50 = 89000 nM T46526 CM75WB 142590122 IC50 = 3700 nM T46526 CM3GL7 142590135 IC50 = 3400 nM T46526 C0H3YO 142590169 IC50 = 1600 nM T46526 CASW65 142590178 IC50 = 44000 nM T46526 C4LG8R 142590181 IC50 = 1600 nM T46526 C7VF5E 142590201 IC50 = 630 nM T46526 C4SO6V 142590222 IC50 = 1500 nM T46526 C8X1QV 142590227 IC50 = 3900 nM T46526 CB04QO 142590230 IC50 = 3100 nM T46526 CVT3O6 142590283 IC50 = 700 nM T46526 C0HF5Y 142590333 IC50 = 890 nM T46526 CZ2XP8 142590348 IC50 = 230 nM T46526 C7PJV6 146981752 IC50 = 630 nM T46526 COIP40 149439735 IC50 = 1500 nM T46526 CLE50J 150904754 IC50 = 81000 nM T46526 C3ZXV1 152835416 IC50 = 970 nM T46526 C92YMQ 153021877 IC50 = 2000 nM T46526 CJBH98 155510838 IC50 = 370 nM T46526 CD2I5X 155511540 IC50 = 92000 nM T46526 CD8KS2 155512016 IC50 = 88000 nM T46526 CGVR19 155521686 IC50 = 1100 nM T46526 CN40JK 155531590 IC50 = 66000 nM T46526 CI35UX 155531642 IC50 = 77000 nM T46526 CKT5D0 155535029 IC50 = 58000 nM T46526 C6X1PU 155537039 IC50 = 48000 nM T46526 C52VTE 155539686 IC50 = 700 nM T46526 CD6VL4 155555091 IC50 = 2700 nM T46526 CUS3K0 155562241 IC50 = 62000 nM T46526 CF2E5H 155564478 IC50 = 51000 nM T46526 C17VLA 113557 IC50 = 65.6 nM T46526 C94FTN 46838079 IC50 = 10.4 nM T46526 CW5D3K 46838218 IC50 = 33000 nM T46526 C4OCA9 4984739 IC50 = 364 nM T46526 D0GS9E 18950 IC50 = 560000 nM T73495 D00ENY 33032 Ki = 701 nM T73495 D02VKC 3272524 Ki = 11730 nM T73495 D0B0NQ 127894 IC50 = 500 nM T73495 D04XMJ 11249042 Ki = 31750 nM T73495 D0OY1V 133058 IC50 > 30000 nM T73495 COC91V 10255 Ki = 177 nM T73495 C71HJK 220181 IC50 > 100000 nM T73495 C37ROZ 439282 Ki = 270 nM T73495 CC0E1V 447081 Ki = 81 nM T73495 C2BWR8 626468 IC50 = 4000 nM T73495 C1EP3D 2733518 Ki = 4800 nM T73495 CWK7X4 4694356 Ki = 6800 nM T73495 CZ2SK5 5287396 Ki = 1300 nM T73495 C3JXD9 5289518 EC50 = 100 nM T73495 CD71AK 6323174 Ki = 56 nM T73495 C5Z8VG 6324635 Ki = 14 nM T73495 C2L6EK 9807075 Ki = 12 nM T73495 CU09JR 9837067 Ki = 28.9 nM T73495 C8ZU6R 9857805 IC50 = 7600 nM T73495 CO37QF 9858686 IC50 > 30000 nM T73495 C9TLQ4 9861035 Ki = 8 nM T73495 C1NB7U 9883705 IC50 = 72000 nM T73495 CFV31D 9946891 IC50 = 4800 nM T73495 C3MAW7 9947478 IC50 = 30000 nM T73495 CG0WB9 9958244 Ki = 3.8 nM T73495 C02TZU 9966866 IC50 = 3700 nM T73495 CLG54O 9977288 IC50 = 3600 nM T73495 CR8AZ9 9995342 IC50 = 36000 nM T73495 C02XFL 9995343 IC50 = 14000 nM T73495 CV90EY 10001987 IC50 = 2200 nM T73495 CX46UD 10065501 IC50 = 3600 nM T73495 CNFM10 10086617 IC50 = 14000 nM T73495 CAN7X8 10087658 IC50 = 3100 nM T73495 CFK0R5 10091990 IC50 = 2000 nM T73495 CF90NL 10109069 IC50 = 5000 nM T73495 CU9FV4 10109670 IC50 = 2200 nM T73495 C20WCA 10131929 IC50 > 100000 nM T73495 C7Q1MJ 10132082 IC50 = 1200 nM T73495 C0B7NU 10177391 IC50 = 60000 nM T73495 CRJ2T0 10219992 Ki = 32.6 nM T73495 CVJ97I 10222090 IC50 = 21000 nM T73495 CU1GH7 10244671 IC50 = 21000 nM T73495 C0KCB7 10268727 IC50 > 100000 nM T73495 CZ2TN4 10268728 IC50 > 100000 nM T73495 CA9TO2 10294563 IC50 = 6100 nM T73495 CQY46K 10316382 IC50 = 4500 nM T73495 C3YP9J 10319750 IC50 = 4700 nM T73495 C5PD0H 10330442 Ki = 54.4 nM T73495 CJ24TX 10330885 Ki = 85.7 nM T73495 C9D8SO 10334434 IC50 = 10000 nM T73495 CBT1U0 10334760 IC50 > 100000 nM T73495 C1OT5C 10339098 IC50 = 4500 nM T73495 CFKJ76 10352480 Ki = 18500 nM T73495 CH3VA0 10358668 IC50 = 12000 nM T73495 C5A1KF 10358931 IC50 = 1300 nM T73495 C70DPZ 10361570 IC50 > 10000 nM T73495 C4WQ3B 10379845 IC50 = 18000 nM T73495 C7GIJ3 10398361 Ki = 241 nM T73495 C18NKE 10402053 IC50 = 31000 nM T73495 CUF4W1 10402054 IC50 = 88000 nM T73495 CVG20W 10409683 IC50 = 5000 nM T73495 C1N2VM 10420002 Ki > 10000 nM T73495 C57CJK 10429001 IC50 = 29000 nM T73495 CX1V3L 10437436 Ki = 100 nM T73495 C0G7JF 10471277 IC50 = 10000 nM T73495 CTX28O 10474107 IC50 = 12000 nM T73495 CAQ65T 10494266 Ki = 254 nM T73495 C1BP3S 10494920 Ki = 3590 nM T73495 CW1DB8 10515815 Ki = 1190 nM T73495 CA1H6P 10518677 Ki = 58 nM T73495 C6XV7F 10520545 Ki = 131 nM T73495 CN7ET5 10536623 Ki = 160 nM T73495 CXE7F5 10541731 Ki = 26 nM T73495 CPR42C 10559986 Ki = 577 nM T73495 C4TS7W 10585396 Ki = 3606 nM T73495 CK20MI 10588564 Ki = 670 nM T73495 CX1J3W 10588885 Ki = 78 nM T73495 CH8R2Z 10589792 Ki = 284 nM T73495 C71YFN 10592589 Ki = 52 nM T73495 C4BQ9F 10608628 Ki = 831 nM T73495 CUN7I9 10632449 Ki = 161 nM T73495 CQ53LW 10638626 Ki = 32 nM T73495 C46KUE 10680281 Ki = 267 nM T73495 CWTN04 10732079 Ki = 367 nM T73495 C7N5AW 10732793 Ki = 60 nM T73495 CMQZ05 10733581 Ki = 59 nM T73495 C1TRI8 10751988 Ki = 2376 nM T73495 C6A4QO 10758246 Ki = 540 nM T73495 CASX36 10773867 Ki = 307 nM T73495 CO0B4H 10774436 Ki = 21 nM T73495 C6U3FQ 10775370 Ki = 41 nM T73495 CCOE52 10777807 Ki = 337 nM T73495 CXWT28 10777943 Ki = 157 nM T73495 C7CA4P 10778899 Ki = 172 nM T73495 C92QWY 10780042 Ki = 40 nM T73495 C30UTV 10797596 Ki = 11.6 nM T73495 CMUE34 10805132 Ki = 7 nM T73495 CB7R3C 10806437 Ki = 49 nM T73495 C4XFQ3 10831138 Ki = 30 nM T73495 CQA6D3 10846340 Ki = 1015 nM T73495 C4G9SI 10854556 Ki = 133 nM T73495 CR5XS2 11153198 Ki = 1200 nM T73495 CRS35K 11154806 Ki = 7370 nM T73495 CQ7E6I 11162637 IC50 = 20000 nM T73495 CLDZ06 11163590 IC50 > 3000 nM T73495 CRA6T3 11175144 IC50 = 31000 nM T73495 CA83CR 11199813 Ki = 800 nM T73495 CQ38WM 11219775 Ki = 5450 nM T73495 CXD0N6 11267855 IC50 = 10000 nM T73495 C8XNV3 11280757 IC50 > 30000 nM T73495 CGRT02 11288627 Ki = 2920 nM T73495 CS3YN5 11302847 IC50 > 3000 nM T73495 C76YPT 11303218 IC50 > 30000 nM T73495 CF58DN 11349236 IC50 > 3000 nM T73495 CZB3R4 11393185 IC50 = 4700 nM T73495 CSYZ37 11395043 IC50 = 12000 nM T73495 CL5T2D 11406465 IC50 > 30000 nM T73495 CBLA18 11415238 IC50 = 51000 nM T73495 CWV6S2 11428576 IC50 > 50000 nM T73495 C9AM3D 11449212 IC50 = 69000 nM T73495 CFR16Q 11452297 IC50 > 30000 nM T73495 C5QT6I 11461651 IC50 = 1200 nM T73495 C8V4UC 11544633 IC50 = 680 nM T73495 CP25TK 11739445 IC50 > 10000 nM T73495 C3NV6L 11742032 IC50 = 1500 nM T73495 C7SHB1 11745400 Ki = 123 nM T73495 CI41BH 11772197 IC50 = 9400 nM T73495 CS26OI 11774516 IC50 > 30000 nM T73495 C06UPV 11791928 Ki = 254 nM T73495 CHUX80 11818375 Ki = 34200 nM T73495 CDGZ79 11820131 Ki = 93.6 nM T73495 CM9WF2 15347043 Ki = 2200 nM T73495 C6AYD8 15347044 Ki = 60.5 nM T73495 C7ES3B 15839907 Ki = 44 nM T73495 CYE1O2 18395300 Ki = 3620 nM T73495 CUP4K1 18944678 IC50 = 12000 nM T73495 CLRK62 22097088 Ki = 530 nM T73495 C0YK6J 22100077 Ki = 330 nM T73495 CM9D7U 22100122 Ki = 230 nM T73495 CJ8UB0 22100152 Ki = 230 nM T73495 CIG65E 22449297 Ki = 1400 nM T73495 C1OW7A 24755637 IC50 = 3.8 nM T73495 CFLR45 24850230 IC50 = 1.9 nM T73495 C0F8KD 44296355 Ki = 152 nM T73495 CY4KI5 44296375 Ki = 224 nM T73495 C0WZ7J 44296493 Ki = 236 nM T73495 C7JD6F 44296494 Ki = 470 nM T73495 C0Y8NC 44296575 Ki > 1000 nM T73495 CI9XM2 44296576 Ki = 150 nM T73495 C6KCR4 44296585 Ki = 29100 nM T73495 CX6LM7 44296601 Ki = 17100 nM T73495 C5LVR2 44296602 Ki = 13900 nM T73495 CJA8X0 44296603 Ki > 1000 nM T73495 CPU32O 44296615 Ki = 41200 nM T73495 CQR8P3 44296800 Ki = 80.4 nM T73495 C2VGB7 44296807 Ki = 6060 nM T73495 C1JV4N 44296812 Ki = 5130 nM T73495 C1RIO8 44296822 Ki = 511 nM T73495 CH3W0P 44301844 Ki = 1464 nM T73495 CJ5X0B 44307207 Ki = 320 nM T73495 C1JC7K 44307264 Ki = 2400 nM T73495 C8U2SF 44307281 Ki = 430 nM T73495 CX8AL2 56945410 IC50 = 650 nM T73495 CDT01W 60023862 Ki = 200 nM T73495 CK7H6W 60023863 Ki = 3200 nM T73495 C86SPH 60023864 Ki = 8000 nM T73495 CJL45I 60023870 Ki = 1100 nM T73495 C0OFZ7 60023874 Ki = 900 nM T73495 CB5X4L 60023875 Ki = 2900 nM T73495 CD54OC 68586104 Ki = 1300 nM T73495 C5U0FY 68586486 Ki = 3700 nM T73495 CQ2XT7 68588179 Ki = 500 nM T73495 CZ6UN9 68588451 Ki = 2100 nM T73495 C7SBU2 68590056 Ki = 1500 nM T73495 CDNJ51 69972507 Ki = 3600 nM T73495 CT3GH6 72543949 Ki = 200 nM T73495 CY67ZT 72543950 Ki = 1100 nM T73495 C10GMK 72544188 Ki = 12800 nM T73495 CMG1J3 72544190 Ki = 900 nM T73495 C7S2RQ 72544191 Ki = 400 nM T73495 C76VSM 72544192 Ki = 10700 nM T73495 CQ90OK 72544193 Ki = 1100 nM T73495 CT30EV 72544414 Ki = 1400 nM T73495 C92PSD 72544415 Ki = 100 nM T73495 CYO4F3 72544417 Ki = 422000 nM T73495 C1HK0F 72544419 Ki = 1000 nM T73495 C0ARY4 72544635 Ki = 700 nM T73495 C3F0SH 72544637 Ki = 20 nM T73495 C2KTJ7 72544639 Ki = 900 nM T73495 CRI79J 72544641 Ki = 90 nM T73495 C91VEK 72544642 Ki = 10000 nM T73495 CHM5L1 72544859 Ki = 900 nM T73495 CRT02N 72544861 Ki = 17000 nM T73495 CD14GW 72544863 Ki = 160 nM T73495 C3W2SA 72544865 Ki = 160 nM T73495 C3EBZ6 72544866 Ki = 1700 nM T73495 CXG0P9 72546282 Ki = 528000 nM T73495 CE6ST8 72546283 Ki = 800 nM T73495 C3B8TH 72546523 Ki = 46000 nM T73495 C3Z1PE 72546524 Ki = 19000 nM T73495 CXWI86 72546765 Ki = 3600 nM T73495 CUJ9A3 72547031 Ki = 2300 nM T73495 C2BEW8 72547032 Ki = 6000 nM T73495 CCO6B5 72547033 Ki = 267000 nM T73495 CZB27J 72547288 Ki = 9700 nM T73495 CVKD75 72547289 Ki = 9900 nM T73495 CBH2X5 72547290 Ki = 19000 nM T73495 CA21EV 72547291 Ki = 11000 nM T73495 CKNW59 72547534 Ki = 5900 nM T73495 CWSJ60 72547535 Ki = 6200 nM T73495 C1DTV4 72547536 Ki = 316000 nM T73495 C6JZ4H 72547537 Ki = 228000 nM T73495 CVID16 73348020 Ki = 67000 nM T73495 CG5PL8 73349560 Ki = 16000 nM T73495 CA2R1Y 76309877 Ki = 3000 nM T73495 CV52YL 76309878 Ki = 600 nM T73495 CJ56PL 135423312 IC50 = 4600 nM T73495 D01RSH 4323128 IC50 = 19000 nM T73495 D03NDD 9935648 Ki = 50 nM T73495 D03RGP 1221 Ki = 740 nM T73495 D0B2VW 95883 Ki = 3 nM T73495 D0K6AF 9839436 Ki = 0.74 nM T73495 D0N1CL 9799478 IC50 = 4800 nM T73495 D0T1MK 656723 Ki = 17130 nM T73495 D0T5SU 158397 Ki = 1150 nM T73495 D0TT9H 4359312 IC50 = 1600 nM T09960 D0NR6S 3002977 IC50 = 1.3 nM T09960 D00XBC 46861584 IC50 = 6309.57 nM T09960 D09JLI 3009355 IC50 = 1.2 nM T09960 D0F7PZ 53316710 IC50 < 0.1 nM T09960 D0O2XQ 11256587 IC50 > 10000 nM T09960 D0O9UC 5275766 IC50 = 3.5 nM T09960 D0Y7NA 49871007 IC50 = 3.1 nM T09960 D0YQ7U 11285792 IC50 = 3 nM T09960 D07GIB 11614352 IC50 = 0.26 nM T09960 D0G6JE 9574343 Ki = 2.1 nM T09960 D0G6SZ 3001322 IC50 = 5.623 nM T09960 D0Q2JS 10436045 Ki = 4260 nM T09960 D0W0LS 183789 IC50 = 1.2 nM T09960 C7Y8VS 1318 EC50 = 4900 nM T09960 CB4Z9P 1474 EC50 = 19000 nM T09960 C78GSK 14338 EC50 = 11000 nM T09960 CW6J7R 15664 EC50 = 2300 nM T09960 CBX47E 20445 IC50 = 501187.23 nM T09960 CD72TB 65237 EC50 = 63095.73 nM T09960 CF1UA4 70848 IC50 = 25000 nM T09960 CR15FN 72791 EC50 > 1000000 nM T09960 C8SC9N 72792 EC50 = 2511.89 nM T09960 C7SIE4 74265 EC50 = 1000 nM T09960 CMJ4V7 77524 EC50 < 1000000 nM T09960 CGZ1C6 77865 EC50 < 1000000 nM T09960 CBW4N5 93149 EC50 = 1800 nM T09960 CTUE81 336912 IC50 = 587000 nM T09960 C2P3FM 353741 IC50 = 199526.23 nM T09960 CW39FG 455656 Ki = 31 nM T09960 C91RPQ 455657 Ki = 32 nM T09960 CLU42H 456292 Ki = 18 nM T09960 CJKB92 456293 Ki = 28 nM T09960 C2K7SR 456298 Ki = 62 nM T09960 CG48QX 456319 IC50 = 90 nM T09960 CN37SU 456323 Ki = 5 nM T09960 C9RGE7 456339 Ki = 15 nM T09960 C70ZGM 456372 Ki = 5 nM T09960 CSOT95 456374 IC50 = 255 nM T09960 CDCZ30 456375 Ki = 1 nM T09960 C4AW8L 456611 Ki = 44 nM T09960 C2VJ3Z 456615 IC50 = 440 nM T09960 CC02UF 456647 Ki = 30 nM T09960 CP3R6C 457671 Ki = 54 nM T09960 CPK6B5 457672 Ki = 29 nM T09960 CNU94V 457679 IC50 = 200 nM T09960 CH6J1S 457797 IC50 > 1000 nM T09960 C42WYA 457829 IC50 > 1000 nM T09960 C9D5BT 457845 IC50 = 980 nM T09960 C78ICG 457871 IC50 = 0.5 nM T09960 C43TRB 457874 Ki = 11 nM T09960 CTU5D6 457875 Ki = 58 nM T09960 C2FHD7 461327 Ki = 5 nM T09960 C8FQ6Y 461546 Ki = 440 nM T09960 CUWT43 461838 Ki = 230 nM T09960 C38ERL 461871 Ki = 45 nM T09960 CHG02J 462395 Ki = 2.7 nM T09960 CR64WQ 462409 Ki = 7 nM T09960 CU43EI 462571 Ki = 10 nM T09960 C47MIH 462573 Ki = 5.23 nM T09960 CKI1S3 462772 Ki = 49 nM T09960 C9YW6M 462902 Ki = 20 nM T09960 CCHZ81 462989 Ki = 18 nM T09960 CF8X4A 463209 Ki = 11 nM T09960 CNVX67 463210 Ki = 11 nM T09960 C2HB4T 463319 Ki = 12 nM T09960 CC85IE 463493 Ki > 1300 nM T09960 C2T0PC 463502 Ki = 74 nM T09960 CH61SC 463517 Ki = 442 nM T09960 C8UQ6H 463616 Ki = 0.7 nM T09960 CVQ5L9 463892 Ki = 11 nM T09960 CAP7I1 464036 Ki = 2 nM T09960 CU29RH 471179 IC50 = 35 nM T09960 C2P0CD 473081 IC50 = 480 nM T09960 C0P7LR 473305 IC50 = 152 nM T09960 CTB56C 474188 Ki = 38 nM T09960 CZ49VF 474465 Ki = 352 nM T09960 CSF9B6 478296 IC50 = 35 nM T09960 CWC96R 478302 IC50 = 30 nM T09960 CRW43A 478307 IC50 = 30 nM T09960 CRF63Q 478308 IC50 = 120 nM T09960 CTF02S 478387 IC50 = 60 nM T09960 C4CD1U 478399 IC50 = 260 nM T09960 C7MVA1 478409 IC50 = 200 nM T09960 CZFM52 478410 IC50 = 25 nM T09960 C2XZ0N 478412 IC50 = 70 nM T09960 CS1NU8 478413 IC50 = 650.13 nM T09960 CTK7B5 478414 IC50 = 50 nM T09960 C0HPV2 478418 IC50 = 120.23 nM T09960 C40OJQ 478439 IC50 = 120.23 nM T09960 C9RM0U 478440 IC50 = 100 nM T09960 C84EFC 478444 IC50 = 4 nM T09960 C6DU8Z 478445 IC50 = 2.5 nM T09960 C79FCT 478446 IC50 = 6 nM T09960 C7BKL5 478447 IC50 = 75 nM T09960 CP60TK 478448 IC50 = 20 nM T09960 CA90RU 478449 IC50 = 100 nM T09960 CC91KL 478450 IC50 = 3.02 nM T09960 C67UKD 478451 IC50 = 3.981 nM T09960 C35VTN 478452 IC50 = 19.95 nM T09960 CF43WD 478471 IC50 > 10000 nM T09960 C1G8DT 478475 IC50 > 10000 nM T09960 CL2CY9 478493 IC50 = 340 nM T09960 CD7NT2 478494 IC50 = 850 nM T09960 CV82HX 478495 IC50 = 1400 nM T09960 CX6WB9 478496 IC50 = 100 nM T09960 C76GKH 478499 IC50 = 70 nM T09960 CP67RF 478500 IC50 = 40 nM T09960 CJ0M6N 478501 IC50 = 150 nM T09960 C0R4CK 478502 IC50 = 60 nM T09960 CH1P4S 478503 IC50 = 40 nM T09960 CPXW62 478508 IC50 > 4000 nM T09960 C2N0BX 478512 IC50 = 340 nM T09960 C10YWE 479835 IC50 = 450 nM T09960 C7TG2M 479837 IC50 = 2000 nM T09960 C2TSP5 479838 IC50 = 1300 nM T09960 CHK75U 479846 IC50 = 90 nM T09960 CE57HZ 479847 IC50 = 110 nM T09960 CQW7Z2 479852 IC50 = 180 nM T09960 CEWR08 479853 IC50 = 110 nM T09960 CW79PV 479855 IC50 > 1000 nM T09960 C8IQ7L 479856 IC50 > 1000 nM T09960 CCHZ69 479857 IC50 = 3000 nM T09960 CR8TC2 479858 IC50 = 100 nM T09960 CVO0B9 479859 IC50 = 110 nM T09960 CT3V4Z 479860 IC50 = 500 nM T09960 CDPW28 479861 IC50 > 1000 nM T09960 C89LZS 479863 IC50 ~ 10000 nM T09960 CR1F7T 479864 IC50 ~ 1000 nM T09960 C0W1KP 479865 IC50 = 200 nM T09960 CEUX01 479866 IC50 > 1000 nM T09960 CBY3Z7 479867 IC50 = 300 nM T09960 C8IMJ5 479868 IC50 = 160 nM T09960 CJ6R0N 479870 IC50 = 570 nM T09960 C8GE2D 479871 IC50 = 60 nM T09960 CKI69Y 479872 IC50 = 180 nM T09960 CX5T0U 479873 IC50 = 110 nM T09960 CAX24K 479874 IC50 > 1000 nM T09960 CCF3N1 479876 IC50 = 400 nM T09960 CJC18Q 479877 IC50 = 100 nM T09960 C6R8FZ 479878 IC50 ~ 10000 nM T09960 C5WRD1 479879 IC50 > 10000 nM T09960 C6OQ5C 479883 IC50 = 80 nM T09960 CT78SG 482147 IC50 = 100 nM T09960 CMZ6P3 482148 IC50 = 50 nM T09960 C35QRN 482150 IC50 = 300 nM T09960 COIA12 482217 IC50 ~ 10000 nM T09960 CKIZ45 483330 IC50 = 15 nM T09960 C6XI2W 483331 IC50 = 27 nM T09960 C4YDE0 483332 IC50 = 111 nM T09960 CCN9V1 483333 IC50 = 335 nM T09960 CAE58G 483334 IC50 = 23 nM T09960 CKU10W 483335 IC50 = 15 nM T09960 C57XVT 483336 IC50 = 15 nM T09960 CN5F7J 483337 IC50 = 16 nM T09960 C7K9DZ 483338 IC50 = 28 nM T09960 CQ3KO7 483339 IC50 = 25 nM T09960 C7AP9W 483340 IC50 = 4 nM T09960 CAB79M 483341 IC50 = 246 nM T09960 C7XW2D 483342 IC50 = 48 nM T09960 C7PMT6 483343 IC50 = 112 nM T09960 CP25RI 483344 IC50 = 10 nM T09960 C9XV0W 483345 IC50 = 18 nM T09960 CDXH14 483348 IC50 = 8600 nM T09960 C6XJ4V 483350 IC50 = 88000 nM T09960 C39BFX 483351 IC50 = 7200 nM T09960 C1T3LZ 483352 IC50 = 24000 nM T09960 CE71IM 483353 IC50 = 4400 nM T09960 C9SUH2 483354 IC50 = 6800 nM T09960 C17BMC 483355 IC50 = 3800 nM T09960 CY7TI4 483356 IC50 = 11000 nM T09960 C1NGQ0 483360 IC50 = 15000 nM T09960 C78PDK 483361 IC50 = 2300 nM T09960 C1FAV4 483362 IC50 = 10400 nM T09960 CI01WP 483363 IC50 = 3500 nM T09960 CH3AK8 483364 IC50 = 8400 nM T09960 CVQG07 483369 IC50 = 1.5 nM T09960 C9SAP8 483382 IC50 = 2 nM T09960 C6EP7Q 483407 EC50 = 1 nM T09960 CN2M0Z 483741 Ki = 590 nM T09960 CTO42Z 483744 Ki = 20 nM T09960 C1TRZ6 483746 Ki = 1300 nM T09960 C4J8NF 483747 IC50 = 0.01 nM T09960 C6E4JZ 484577 Ki = 5 nM T09960 CBLP57 484578 Ki = 3 nM T09960 CQX89C 484579 Ki = 5 nM T09960 C2PZO7 484581 Ki = 8 nM T09960 CAXL81 486595 IC50 = 400 nM T09960 C8KY2N 486601 IC50 = 2 nM T09960 CC17IT 486602 IC50 = 4 nM T09960 CUJ4P3 486604 IC50 = 1.5 nM T09960 C1F4ZP 486605 IC50 = 0.8 nM T09960 C7UVY2 486606 IC50 = 2 nM T09960 CTG0K5 486607 IC50 = 3 nM T09960 C0N1KQ 486608 IC50 = 120 nM T09960 CT8JO0 486632 IC50 = 1.5 nM T09960 CP6ZN1 489305 IC50 = 6.5 nM T09960 C64KTB 489306 IC50 = 3 nM T09960 C97FKT 489307 IC50 = 4 nM T09960 C6EAD2 489308 IC50 = 2 nM T09960 CD9CA1 489312 IC50 = 25 nM T09960 C0GS3N 489313 IC50 = 41 nM T09960 CL5UD4 489314 IC50 = 60 nM T09960 CHUB62 489315 IC50 = 0.3 nM T09960 C90YRJ 489316 IC50 = 6.5 nM T09960 C91OWI 489593 IC50 > 10000 nM T09960 C7QDT0 489594 IC50 = 26 nM T09960 C9Q8MV 489595 IC50 = 49 nM T09960 CFZ02X 489596 IC50 > 10000 nM T09960 CP15BS 489597 IC50 = 3500 nM T09960 CZ39NR 489598 IC50 > 10000 nM T09960 CWM08J 489599 IC50 > 10000 nM T09960 C6AD2R 489805 IC50 = 610 nM T09960 CLB6T9 489806 IC50 = 67 nM T09960 C03VWO 489807 IC50 = 155 nM T09960 CVR7Q0 489808 IC50 = 52 nM T09960 C4HO2V 489809 IC50 = 94 nM T09960 CBO93F 489810 IC50 = 750 nM T09960 CRXG81 489811 IC50 = 140 nM T09960 CO7AN1 489812 IC50 = 140 nM T09960 CLU42C 489813 IC50 > 1000 nM T09960 C6BLV4 489814 IC50 = 97 nM T09960 C7XR9V 489815 IC50 = 96 nM T09960 C04MOK 489816 IC50 = 89 nM T09960 C38MNQ 489817 IC50 = 48 nM T09960 CWP0O9 489818 IC50 = 32 nM T09960 CBGQ95 489820 IC50 = 260 nM T09960 CR78CU 489821 IC50 = 55 nM T09960 CS3Q6D 489822 IC50 = 46 nM T09960 CM78TR 489823 IC50 = 33 nM T09960 CK25FT 489824 IC50 = 34 nM T09960 CXV7H5 489825 IC50 = 19 nM T09960 CJQF51 489826 IC50 = 48 nM T09960 CLB51I 489827 IC50 = 57 nM T09960 C4WES0 489828 IC50 > 1000 nM T09960 CNU5F6 489829 IC50 = 810 nM T09960 C20OGE 489830 IC50 > 1000 nM T09960 C6L0XZ 489831 IC50 > 1000 nM T09960 CG24QV 489832 IC50 > 1000 nM T09960 CE09IT 489833 IC50 = 390 nM T09960 CYA56U 489834 IC50 > 1000 nM T09960 C9K7VD 489835 IC50 = 150 nM T09960 CA4KS9 490006 IC50 = 46 nM T09960 CIYP51 490007 IC50 = 31 nM T09960 C8OH9Y 490008 IC50 = 12 nM T09960 C8MH9R 490010 IC50 = 17 nM T09960 C1ZY4G 490011 IC50 = 15 nM T09960 C7QR3K 490012 IC50 = 9 nM T09960 C7PF8H 490013 IC50 = 5 nM T09960 CBG64R 490014 IC50 = 2 nM T09960 CQZW31 490016 IC50 = 4 nM T09960 C15GOK 490017 IC50 = 2 nM T09960 CV06XI 490018 IC50 = 0.1 nM T09960 C9YNU2 490019 IC50 = 0.2 nM T09960 CP8MR9 490020 IC50 = 0.8 nM T09960 C4R0QW 490022 IC50 = 0.8 nM T09960 C3PH6B 490023 IC50 = 0.2 nM T09960 CA5BZ8 491773 IC50 = 38 nM T09960 C9NE3B 496970 IC50 = 100 nM T09960 CI7GR8 496971 IC50 = 3 nM T09960 CJVQ67 496972 IC50 = 10 nM T09960 CQKL02 496973 IC50 = 5.998 nM T09960 CZ0W8A 496974 IC50 = 5 nM T09960 C6EDZ1 496975 IC50 = 2 nM T09960 C5BP9E 496983 IC50 = 6.998 nM T09960 CZ67QC 496984 IC50 = 5.998 nM T09960 CN9OE4 496985 IC50 = 12 nM T09960 C5HGF3 501043 IC50 = 1 nM T09960 CU4R2W 501044 IC50 = 3.6 nM T09960 C1GA2L 501045 IC50 = 1 nM T09960 CQ38YL 501046 IC50 = 0.5 nM T09960 C7TYW3 501047 IC50 = 1 nM T09960 C0YM7T 501048 IC50 = 24 nM T09960 C3GTE7 501049 IC50 = 4 nM T09960 CSYH30 501050 IC50 = 5 nM T09960 C2XT8B 501051 IC50 = 0.7998 nM T09960 CUR04D 501052 IC50 = 2 nM T09960 CGD5I0 501053 IC50 = 3 nM T09960 C6YVK3 501054 IC50 = 5.998 nM T09960 CZYS12 501055 IC50 = 0.1 nM T09960 C0L6BS 501056 IC50 = 0.7 nM T09960 CR3K8B 501057 IC50 = 3.999 nM T09960 C4R8TH 501058 IC50 = 36 nM T09960 CWL94S 501059 IC50 = 3 nM T09960 C4EYK5 501060 IC50 = 0.1 nM T09960 CP8ON7 501062 IC50 = 0.1 nM T09960 C0Y7TL 501063 IC50 = 0.2 nM T09960 C7JQ2Z 502259 Ki = 10 nM T09960 C9N6LP 503637 Ki = 5.1 nM T09960 CN7P0G 505865 IC50 = 300 nM T09960 CSAM47 505866 IC50 = 9 nM T09960 C40MHP 505867 IC50 = 10 nM T09960 C3WXP0 505868 IC50 = 12 nM T09960 CF8TK4 505869 IC50 = 6 nM T09960 CZ0KC5 505870 IC50 = 9 nM T09960 C2A1QX 505873 IC50 = 12 nM T09960 C15FCB 505874 IC50 = 66 nM T09960 C43SIR 505875 IC50 = 12 nM T09960 CQ9S3K 505876 IC50 = 42 nM T09960 CSZ3V1 505878 IC50 = 3.9 nM T09960 CJ24LQ 505879 IC50 = 5 nM T09960 CSIQ81 505880 IC50 = 6.6 nM T09960 CJ4P1O 505881 IC50 = 1.6 nM T09960 CD09FO 511294 Ki = 68 nM T09960 CZHY61 511295 Ki = 110 nM T09960 CC0WK3 511296 Ki = 86 nM T09960 C2YCQ4 511297 Ki = 360 nM T09960 CS61JO 511298 Ki = 190 nM T09960 CQE5N9 511299 Ki = 62 nM T09960 CN25FS 511303 Ki = 33 nM T09960 COCZ64 511304 Ki = 25 nM T09960 C2Z4CB 511305 Ki = 55 nM T09960 CU5DY2 511306 Ki = 155 nM T09960 CPW6C4 511307 Ki = 33 nM T09960 CC70RW 511308 Ki = 596 nM T09960 C1YFM7 511309 Ki = 8 nM T09960 CFJ63U 511332 Ki = 7 nM T09960 C49UTP 516172 IC50 = 1.199 nM T09960 CFY12E 516173 IC50 = 1.5 nM T09960 C17QUG 516174 IC50 = 2.3 nM T09960 CE7IZ3 516175 IC50 = 1.1 nM T09960 CAK7I5 516176 IC50 = 1.3 nM T09960 CJKA08 516177 IC50 = 2.2 nM T09960 CJ10ZD 516178 IC50 = 1.1 nM T09960 CLNW94 516179 IC50 = 2.6 nM T09960 C36DAX 516180 IC50 = 5 nM T09960 C17OWX 516181 IC50 = 1.3 nM T09960 CTR8J0 516182 IC50 = 2 nM T09960 CIT5M7 516183 IC50 = 3.2 nM T09960 CWI3S4 516184 IC50 = 3.1 nM T09960 C9H8KU 516185 IC50 = 1.7 nM T09960 C5XTV2 516186 IC50 = 3.5 nM T09960 C8AEM1 516187 IC50 = 1.3 nM T09960 CPE45H 516188 IC50 = 13.1 nM T09960 CF2ER3 516189 IC50 = 1.3 nM T09960 CZDN60 516190 IC50 = 1 nM T09960 C19ZRH 516191 IC50 = 0.8 nM T09960 C3VUY8 516192 IC50 = 0.5 nM T09960 C2UA5G 516193 IC50 = 1 nM T09960 C68PSM 516194 IC50 = 0.6 nM T09960 C2U3FJ 516195 IC50 = 0.8 nM T09960 C8T4PC 516196 IC50 = 0.6 nM T09960 C02BWL 516197 IC50 = 0.8 nM T09960 CA3W8V 516198 IC50 = 0.5 nM T09960 CICH26 516199 IC50 = 0.6 nM T09960 CQ1PG6 516200 IC50 = 0.8 nM T09960 CKI1J9 516201 IC50 = 0.4 nM T09960 CUX94K 516202 IC50 = 0.3 nM T09960 CNCR59 516203 IC50 = 0.9 nM T09960 C3A9RP 516204 IC50 = 1.2 nM T09960 CN80KP 516205 IC50 = 0.5 nM T09960 CTAR48 516206 IC50 = 2.1 nM T09960 C4Y1EX 516207 IC50 = 1.3 nM T09960 CMH39L 516208 IC50 = 0.9 nM T09960 CXD32U 516209 IC50 = 0.6 nM T09960 CB0PW1 516211 IC50 = 1.2 nM T09960 C9MVL1 516212 IC50 = 0.6 nM T09960 C2ISE5 516213 IC50 = 0.9 nM T09960 CBEO51 516214 IC50 = 1.1 nM T09960 CR15ZC 516215 IC50 = 1 nM T09960 CNSQ90 516216 IC50 = 0.3 nM T09960 CJUT37 516217 IC50 = 1.3 nM T09960 CMZ6C3 516218 IC50 = 0.8 nM T09960 C1F7HO 516219 IC50 = 1.3 nM T09960 C7SLM0 516220 IC50 = 0.7 nM T09960 CRD07L 516221 IC50 = 0.4 nM T09960 C97TAX 516222 IC50 = 1.1 nM T09960 CRG4W0 516223 IC50 = 0.6 nM T09960 C4BX1V 516224 IC50 = 0.3 nM T09960 CE1DA2 516225 IC50 = 1.4 nM T09960 C2WHI5 516226 IC50 = 1.5 nM T09960 CJ7E9S 516227 IC50 = 0.5 nM T09960 C23VSR 516228 IC50 = 0.5 nM T09960 C70EVZ 516229 IC50 = 0.7 nM T09960 CC8HS5 516230 IC50 = 0.4 nM T09960 CJ02LM 516231 IC50 = 0.3 nM T09960 CK1U5W 516232 IC50 = 0.3 nM T09960 C9UOI0 516233 IC50 = 0.3 nM T09960 C5D1XY 516234 IC50 = 0.3 nM T09960 C67BKT 516235 IC50 = 0.3 nM T09960 CL2KZ5 516236 IC50 = 0.9 nM T09960 CW9M7J 516237 IC50 = 0.5 nM T09960 CDTJ57 516238 IC50 = 1.6 nM T09960 CWTN29 516239 IC50 = 1.3 nM T09960 C0CAK2 516240 IC50 = 1.1 nM T09960 CV6JB5 516241 IC50 = 2.7 nM T09960 C4MG1X 516242 IC50 = 0.8 nM T09960 CGT3M2 516243 IC50 = 1.2 nM T09960 CM4D9P 516244 IC50 = 0.8 nM T09960 C4HF7G 516245 IC50 = 0.3 nM T09960 C6L1BX 516246 IC50 = 0.4 nM T09960 C4MQR0 516247 IC50 = 1.6 nM T09960 CK64CJ 516248 IC50 = 0.5 nM T09960 C1MP9U 516249 IC50 = 0.5 nM T09960 CA0CL5 516250 IC50 = 0.6 nM T09960 CIOG73 516251 IC50 = 0.5 nM T09960 CHZ03N 516252 IC50 = 0.6 nM T09960 CSWV89 516253 IC50 = 0.6 nM T09960 C1LB4X 516254 IC50 = 2.6 nM T09960 CA02XT 516255 IC50 = 0.4 nM T09960 CI76WJ 516256 IC50 = 0.2 nM T09960 C8SLJ6 516257 IC50 = 0.2 nM T09960 C5JO7X 516258 IC50 = 0.8 nM T09960 C1ZBU6 516259 IC50 = 0.5 nM T09960 CQ52IA 516260 IC50 = 0.7998 nM T09960 CJ71SM 516261 IC50 = 1.1 nM T09960 CDSF01 516262 IC50 = 0.3 nM T09960 CBEN83 516263 IC50 = 2.3 nM T09960 C65AZI 516264 IC50 = 1.3 nM T09960 CVK8R9 516266 IC50 = 1.6 nM T09960 C4Z1UM 516267 IC50 = 1.1 nM T09960 CCD9S6 516268 IC50 = 1.5 nM T09960 C72UXL 516269 IC50 = 0.7 nM T09960 CMJZ98 516270 IC50 = 0.9 nM T09960 C3ORY7 516271 IC50 = 0.4 nM T09960 CUB96H 516272 IC50 = 0.8 nM T09960 C86FJD 516273 IC50 = 0.8 nM T09960 C8JI6P 516274 IC50 = 0.4 nM T09960 COA04U 516275 IC50 = 0.7 nM T09960 C59YWP 516276 IC50 = 0.7 nM T09960 C75MOZ 516277 IC50 = 2 nM T09960 CIJX71 516278 IC50 = 1.1 nM T09960 C8ZT2N 516279 IC50 = 0.4 nM T09960 C9XU6R 516280 IC50 = 0.6 nM T09960 CSU21I 516281 IC50 = 0.6 nM T09960 CA56QB 516282 IC50 = 0.5 nM T09960 C28OFN 516283 IC50 = 1.1 nM T09960 CHN28A 516284 IC50 = 1.2 nM T09960 C8DAC7 516285 IC50 = 0.7 nM T09960 C5L4MQ 516286 IC50 = 0.9 nM T09960 CJ8NY1 516287 IC50 = 0.7 nM T09960 CY1B6X 516288 IC50 = 0.2 nM T09960 C1I4UL 516289 IC50 = 0.2 nM T09960 CK93QH 516290 IC50 = 0.6 nM T09960 CFKI94 516291 IC50 = 0.6 nM T09960 CBYO78 516292 IC50 = 0.4 nM T09960 C4XN2D 516293 IC50 = 0.6 nM T09960 C9D5QE 516294 IC50 = 1.6 nM T09960 CN8XA2 516295 IC50 = 1.1 nM T09960 CK1PD5 516296 IC50 = 1 nM T09960 CFEW91 516298 IC50 = 0.9 nM T09960 CDMW14 516299 IC50 = 1.5 nM T09960 C97KFD 516300 IC50 = 0.9 nM T09960 CBXT91 516301 IC50 = 1.5 nM T09960 CI5Q8L 516302 IC50 = 1.7 nM T09960 C8L2AF 516303 IC50 = 2.3 nM T09960 C8J2GI 516304 IC50 = 0.8 nM T09960 C2I3NA 516305 IC50 = 3.9 nM T09960 CN7MX3 516306 IC50 = 1.1 nM T09960 CZ23TX 516307 IC50 = 1 nM T09960 C6K0JX 516308 IC50 = 0.7 nM T09960 CL3P0C 516309 IC50 = 0.8 nM T09960 CV7JI2 516310 IC50 = 0.2 nM T09960 C81OXC 516311 IC50 = 0.5 nM T09960 C95XCF 516312 IC50 = 0.5 nM T09960 CNZ5I9 516313 IC50 = 0.5 nM T09960 CUAO78 516314 IC50 = 0.3 nM T09960 CG02IZ 516315 IC50 = 76 nM T09960 C1A0SH 516319 IC50 = 78 nM T09960 C92CLD 516325 IC50 = 2.198 nM T09960 C5Z9TB 516326 IC50 = 4.2 nM T09960 C3C0IU 516327 IC50 = 4.6 nM T09960 C0H9RE 516328 IC50 = 2.999 nM T09960 C8KPC3 516329 IC50 = 4.8 nM T09960 C3F0MY 516330 IC50 = 9 nM T09960 CUK2G8 516331 IC50 = 33 nM T09960 CGB36E 516332 IC50 = 2.999 nM T09960 CCJ4U8 516333 IC50 = 0.6 nM T09960 CAK2S5 516334 IC50 = 4.8 nM T09960 C8R5IX 516335 IC50 = 1.2 nM T09960 CK70CG 516336 IC50 = 1 nM T09960 CB14VJ 516337 IC50 = 0.6 nM T09960 COA15S 516338 IC50 = 20 nM T09960 CD8S9J 516339 IC50 = 2.3 nM T09960 C16UMB 516340 IC50 = 23 nM T09960 CQE9N8 516341 IC50 = 9 nM T09960 C7WHX0 516342 IC50 = 0.7998 nM T09960 C1EJM4 516343 IC50 = 1.199 nM T09960 CM1QB4 516344 IC50 = 22 nM T09960 CJ0BW8 516345 IC50 = 16 nM T09960 CZ54ST 516346 IC50 = 121.9 nM T09960 C8W3IM 516347 IC50 = 7.5 nM T09960 CDE5F0 516348 IC50 = 7.5 nM T09960 CF29PH 516349 IC50 = 16 nM T09960 C5DHL6 516350 IC50 = 9 nM T09960 CDAS93 516351 IC50 = 4 nM T09960 CH68TF 516352 IC50 = 12 nM T09960 CZ4YM1 516353 IC50 = 2.2 nM T09960 CAX3D4 516354 IC50 = 2.099 nM T09960 CCF0X5 516357 IC50 = 11.5 nM T09960 C1S2KP 516358 IC50 = 6.9 nM T09960 CE6O0T 516361 IC50 = 1.199 nM T09960 CKH2Z9 516362 IC50 = 1.199 nM T09960 CU32RP 516363 IC50 = 2.9 nM T09960 C3GA8B 516364 IC50 = 2.8 nM T09960 CE3FO7 516365 IC50 = 1.6 nM T09960 CNY7F9 516366 IC50 = 0.8995 nM T09960 C5R6OZ 516367 IC50 = 1.6 nM T09960 CJU93H 516368 IC50 = 5.5 nM T09960 CSF9D4 602123 IC50 = 125892.54 nM T09960 CXMY27 619353 IC50 = 501187.23 nM T09960 CYU56N 667748 IC50 = 8100 nM T09960 CMP4D3 1167892 EC50 = 3000 nM T09960 CAF8P7 2733927 EC50 = 19952.62 nM T09960 C90AHY 3002976 IC50 = 1 nM T09960 C1IPS0 3007227 IC50 = 105 nM T09960 CUY7J9 3008902 IC50 = 2 nM T09960 C1V4TU 3008903 IC50 = 80 nM T09960 CE3Q4V 3008904 IC50 = 2.8 nM T09960 CG7ZT5 3008905 IC50 = 3.8 nM T09960 C6VG7U 3008906 IC50 > 1000 nM T09960 C32FTI 3008907 IC50 = 100 nM T09960 CQR7S5 3008908 IC50 = 2 nM T09960 C8JLB6 3008909 IC50 = 27.3 nM T09960 C45FME 3008910 IC50 = 460 nM T09960 CC23PJ 3008911 IC50 = 102 nM T09960 CR3K2Z 3008912 IC50 = 43 nM T09960 CZ1V8Q 3008913 IC50 = 3 nM T09960 CDSG05 3008914 IC50 = 2.3 nM T09960 C4V0IN 3008915 IC50 > 1000 nM T09960 CKXR32 3008916 IC50 = 75 nM T09960 C1IS9G 3008917 IC50 = 0.7 nM T09960 CP12EY 3008918 IC50 = 7.8 nM T09960 CK83ZH 3008919 IC50 = 200 nM T09960 CEX1C8 3008920 IC50 > 100 nM T09960 CUNQ43 3008921 IC50 = 408 nM T09960 CI21SO 3008922 IC50 = 42 nM T09960 CU38DW 3008923 IC50 = 2.4 nM T09960 CI87PX 3008924 IC50 = 3.7 nM T09960 C2IW9S 3008925 IC50 = 31 nM T09960 C0PHV5 3008926 IC50 = 283 nM T09960 CZV0O6 3008927 IC50 = 1.1 nM T09960 C83ZWQ 3008928 IC50 = 1 nM T09960 CHQS14 3008929 IC50 = 3.3 nM T09960 C8KY7B 3008930 IC50 = 2.9 nM T09960 CH3L2R 3008931 IC50 = 16.5 nM T09960 C0JWL6 3008932 IC50 = 2.8 nM T09960 C0N8VX 3008933 IC50 = 41 nM T09960 CK7N8Y 3008934 IC50 = 11.1 nM T09960 CA58WE 3008935 IC50 = 15.5 nM T09960 C36JPC 3008936 IC50 = 9 nM T09960 CGU6O8 3008937 IC50 = 62 nM T09960 CUF0Z9 3009352 Ki = 5.2 nM T09960 CMK58I 3009353 Ki = 1.1 nM T09960 CPN54Q 3009354 Ki = 1.4 nM T09960 C6ZYX5 3009356 Ki = 1.6 nM T09960 CM80UB 3010250 IC50 = 6000 nM T09960 C2PNE4 3010251 IC50 = 6000 nM T09960 CB9C6Y 3010252 IC50 = 15000 nM T09960 CJBC38 3010256 IC50 = 18.1 nM T09960 C7GV5W 3010257 IC50 = 27 nM T09960 CVC2U8 3010258 IC50 = 23 nM T09960 C5XB2T 3010259 IC50 = 6.2 nM T09960 CX9PH2 3010260 IC50 = 1.1 nM T09960 CLR3U2 3010261 IC50 = 0.67 nM T09960 CIS59J 3010262 IC50 = 1.3 nM T09960 CVL16O 3010263 IC50 = 2 nM T09960 CX3IP6 3010264 IC50 = 0.2897 nM T09960 C5WT4G 3010265 IC50 = 1.5 nM T09960 CLSN01 3010266 IC50 = 7 nM T09960 C0DJQ4 3010267 IC50 = 0.73 nM T09960 C1T3CG 3010268 IC50 = 0.38 nM T09960 C7JI2E 3010269 IC50 = 3.802 nM T09960 CKS98E 3010270 IC50 = 1.6 nM T09960 CD16BY 3010271 IC50 = 0.34 nM T09960 C2TG9W 3010272 IC50 = 0.51 nM T09960 CGZV74 3010273 IC50 = 0.23 nM T09960 CC8YU9 3010274 IC50 = 0.23 nM T09960 CA2LX4 3010275 IC50 = 0.57 nM T09960 C7ON3J 3010276 IC50 = 0.6 nM T09960 CJQ5B0 3010277 IC50 = 0.89 nM T09960 CQC1H6 3010278 IC50 = 0.76 nM T09960 C4RFK6 3010279 IC50 = 0.7 nM T09960 CW3OZ1 3010280 IC50 = 1 nM T09960 C0WZ9R 3011719 IC50 = 363 nM T09960 C7SG4P 3011721 IC50 = 83 nM T09960 CFOY69 3011722 IC50 = 339 nM T09960 C5R1AW 3011723 IC50 = 8.9 nM T09960 CF53ZB 3011725 IC50 = 126 nM T09960 CSED31 3011729 IC50 = 5 nM T09960 CWOH42 3011734 IC50 = 2.4 nM T09960 C53JFX 3013575 IC50 = 5.3 nM T09960 CD5LN4 3013673 IC50 = 16 nM T09960 CZSP97 3013684 IC50 = 1.2 nM T09960 C7M4ZG 3013689 IC50 = 2.1 nM T09960 C6AV0J 3013701 IC50 = 0.8 nM T09960 CZ9M6G 3209888 IC50 = 79400 nM T09960 CNK42U 3258407 EC50 = 1900 nM T09960 CZ2G4M 4080740 IC50 = 49000 nM T09960 CKEC40 5275759 IC50 = 1.4 nM T09960 CD3C4L 5275760 IC50 = 4.6 nM T09960 C56OAD 5275761 IC50 = 44 nM T09960 C6N2GA 5275762 IC50 = 8.9 nM T09960 CE52UZ 5275763 IC50 = 5.1 nM T09960 CD9UY7 5275764 IC50 = 8.2 nM T09960 CPH85Y 5275765 IC50 = 2.2 nM T09960 C8RK0Q 5275829 IC50 = 2 nM T09960 CPUL05 5275832 IC50 = 36.7 nM T09960 CSMT51 5275833 IC50 = 350 nM T09960 CMVX10 5275835 IC50 = 11 nM T09960 CCI94R 5275836 IC50 > 2000 nM T09960 CWJC59 5275837 IC50 = 9 nM T09960 C0QK9G 5275839 IC50 = 6.4 nM T09960 CU0IJ1 5275840 IC50 = 28 nM T09960 C7UZ4T 5275841 IC50 = 10 nM T09960 CAT0F3 5275842 IC50 = 5.3 nM T09960 COFC54 5347695 IC50 > 30000 nM T09960 C04WJE 5479787 IC50 = 40 nM T09960 C9LO0F 5479840 Ki = 19 nM T09960 C59FSP 5479841 Ki = 1.1 nM T09960 CGH7F6 5479842 Ki = 3.4 nM T09960 CHXB92 5479843 Ki = 2 nM T09960 CCW7L9 5479844 Ki = 1.8 nM T09960 CQ63MB 5479845 Ki = 2 nM T09960 CS64KP 5479851 Ki = 18 nM T09960 C54DRO 5479852 Ki = 4.5 nM T09960 CMT8K7 5481702 IC50 = 10 nM T09960 C95HGD 5481703 IC50 = 15 nM T09960 CQ1WY9 5481704 IC50 = 100 nM T09960 C6DS7P 5481705 IC50 = 399.94 nM T09960 CF6W1C 5481707 IC50 = 1199.5 nM T09960 CZO76A 5481711 IC50 = 180 nM T09960 CXAK62 5481712 IC50 = 50 nM T09960 CMK83F 5481713 IC50 = 5 nM T09960 C31PZY 5481714 IC50 = 100 nM T09960 CYK98N 5481715 IC50 = 299.92 nM T09960 C7JH1S 5481716 IC50 = 100 nM T09960 CQFS90 5481726 IC50 = 120 nM T09960 C2X7VQ 5481727 IC50 = 699.84 nM T09960 CN95LU 5481736 IC50 = 640 nM T09960 CDGR53 5481737 IC50 = 780 nM T09960 C0L1UR 5481741 IC50 = 1000 nM T09960 CE3MS6 5481742 IC50 = 4 nM T09960 CUCQ49 5481743 IC50 = 4 nM T09960 C9R1OG 5481744 IC50 = 50 nM T09960 C2UG0D 5481745 IC50 = 449.78 nM T09960 C4NP6M 5481746 IC50 = 40 nM T09960 CD8H1T 5481747 IC50 = 2600.16 nM T09960 CTHN69 5481748 IC50 = 60 nM T09960 COU51D 5481749 IC50 = 5902.01 nM T09960 C01YKP 5481750 IC50 = 100 nM T09960 C1BZ4F 5481751 IC50 = 90 nM T09960 C3M6UP 5481752 IC50 = 120 nM T09960 CQTH08 5481754 IC50 = 100 nM T09960 CF5AX1 5481859 IC50 = 270 nM T09960 CD3I2R 5481861 IC50 = 270 nM T09960 C6UZJ0 5481866 IC50 = 200 nM T09960 C3HG0F 5481867 IC50 = 80 nM T09960 CZU13P 5481871 IC50 = 570 nM T09960 C3PTO2 5482298 Ki = 1.1 nM T09960 CF6PQ5 5482299 Ki = 2.2 nM T09960 CAY72C 5482300 Ki = 0.4 nM T09960 CU9D7T 5482301 Ki = 0.3 nM T09960 CSM61O 5482453 IC50 = 35 nM T09960 C6P2SJ 5482454 IC50 = 35 nM T09960 CM4SG8 5482456 IC50 = 2400 nM T09960 CR37LY 5482457 IC50 = 599.79 nM T09960 C5E4PX 5482807 IC50 = 1600 nM T09960 CSDH37 5482808 IC50 = 230 nM T09960 CMG39Z 5482809 IC50 = 10000 nM T09960 C2WV1F 5482810 IC50 = 130 nM T09960 CAY0F1 5482811 IC50 = 160 nM T09960 CLH72E 5495579 Ki = 23 nM T09960 C06TBN 5495580 Ki = 8.8 nM T09960 CZL2A6 5495581 Ki = 1.2 nM T09960 C1CBX6 5495582 Ki = 0.7 nM T09960 CZ34KJ 5495583 Ki = 4.7 nM T09960 CZMA67 5495584 Ki = 2 nM T09960 C73MGH 5495585 Ki = 14 nM T09960 CC32FY 5495586 Ki = 8.1 nM T09960 CB5ZE4 5495587 Ki = 11 nM T09960 C94XKN 5495588 Ki = 3.3 nM T09960 C94XMP 5495589 Ki = 2.1 nM T09960 CSQ6J1 5495590 Ki = 3.2 nM T09960 C3QE4X 5495591 Ki = 5.7 nM T09960 C1FJ2B 5495592 Ki = 60 nM T09960 CCD24B 5495593 Ki = 315 nM T09960 CJ02MD 5495594 Ki = 43 nM T09960 CJ6WT9 5495595 Ki = 25 nM T09960 C72OIB 5495596 Ki = 5.3 nM T09960 C6AIC7 5495597 Ki = 1.3 nM T09960 C8Q2HF 5496098 Ki = 78 nM T09960 CU45LD 5496099 Ki = 3 nM T09960 CCS5G7 5496100 Ki = 9 nM T09960 C6YTS3 5496101 Ki = 4 nM T09960 CGZ4H2 5496102 Ki = 33 nM T09960 C6U1JH 5496103 Ki = 33 nM T09960 CWK9Z7 5496104 Ki > 30 nM T09960 C9EKW0 5496105 Ki = 26 nM T09960 C3K4OF 5496106 Ki > 30 nM T09960 CJ6PF5 5496107 Ki = 7 nM T09960 CD39HS 5496108 Ki = 43 nM T09960 CNV6Y1 5496109 Ki > 30 nM T09960 C2JN1C 5496110 Ki > 30 nM T09960 C6RW0S 5496111 Ki > 30 nM T09960 CPBD91 5496112 Ki = 16 nM T09960 CCDG57 5496113 Ki = 5.3 nM T09960 C65BAI 5496114 Ki = 7.6 nM T09960 C7EQ2H 5496115 Ki = 30 nM T09960 CL9T5D 5496116 Ki = 24 nM T09960 C7QFB3 5496117 Ki = 3.8 nM T09960 C86DKQ 5496118 Ki = 4.4 nM T09960 C1VGC8 5496119 Ki = 20 nM T09960 CETR80 5496120 Ki = 5.6 nM T09960 CWLT23 5496121 Ki = 30 nM T09960 CA74LD 6320546 IC50 = 51 nM T09960 CU64LG 6320579 IC50 = 31.9 nM T09960 CHC9Y0 6320580 IC50 > 100 nM T09960 C2U7CA 6320581 IC50 = 16 nM T09960 CB41ZV 6320582 IC50 = 2 nM T09960 CLY09O 6320585 IC50 = 2 nM T09960 CY3S4K 6480206 IC50 = 32000 nM T09960 C9AFC3 6532433 Ki = 2.2 nM T09960 CD03OA 6532434 Ki = 0.4 nM T09960 CK5F9T 6532435 Ki = 0.3 nM T09960 C7J6DP 6532436 Ki = 0.1 nM T09960 C0IGN3 6533779 Ki = 2.3 nM T09960 C3E9JO 6533780 Ki = 8.8 nM T09960 CJ0I8N 6533781 Ki = 1.2 nM T09960 CHCY06 6918496 IC50 > 1000 nM T09960 C3M8YI 9574356 Ki = 18 nM T09960 CG4WA2 9574357 Ki = 1.1 nM T09960 CJN17G 9574358 Ki = 3.4 nM T09960 C59BRT 9574359 Ki = 18 nM T09960 CD2SY1 9574360 Ki = 4.5 nM T09960 C6C0XH 9575320 Ki = 1.1 nM T09960 C7GYD5 9579116 Ki = 0.7 nM T09960 C68CDO 9579117 Ki = 4.7 nM T09960 C2MV5K 9808628 IC50 = 25 nM T09960 C5T8RE 9809508 IC50 = 4.5 nM T09960 CC5EI0 9810893 IC50 = 0.24 nM T09960 CO1JI7 9827221 IC50 = 6 nM T09960 CY39ML 9869601 IC50 = 199.99 nM T09960 C9FO1Q 9873546 IC50 = 72 nM T09960 COHL06 9894474 IC50 = 240 nM T09960 C46YOP 9909684 IC50 = 6100 nM T09960 CZ7P4T 9914742 IC50 = 1.8 nM T09960 CU5O1J 9915724 IC50 = 19 nM T09960 C03TPL 9916998 IC50 = 0.22 nM T09960 CX9V2G 9917628 IC50 = 1.8 nM T09960 CSH40U 9936494 IC50 = 20 nM T09960 CQ76HK 9938497 IC50 = 43 nM T09960 C91RTG 9956238 IC50 = 400 nM T09960 C0FHY1 9978318 IC50 = 5500 nM T09960 CRP06Q 10008425 IC50 = 7.244 nM T09960 CPXO85 10008490 IC50 = 4786.3 nM T09960 C3VB2C 10008665 IC50 = 2.5 nM T09960 CVG30F 10008921 IC50 = 9120.11 nM T09960 CG1KV2 10030170 IC50 = 3 nM T09960 C1X9CD 10053691 IC50 = 1479.11 nM T09960 C4S1FH 10076141 IC50 = 0.05998 nM T09960 CRT92N 10116073 IC50 = 3000 nM T09960 C49DEF 10117347 IC50 = 120 nM T09960 C2B4CH 10118535 IC50 = 330 nM T09960 C52GKX 10143882 IC50 = 300 nM T09960 C2U4WP 10159217 IC50 = 560 nM T09960 CR2WS1 10163007 IC50 = 0.5 nM T09960 C1BGH8 10182763 IC50 = 7600 nM T09960 C2ED3X 10184169 IC50 = 2000 nM T09960 C4UC7K 10186729 IC50 = 24 nM T09960 C3DM7B 10186910 IC50 = 1.7 nM T09960 C16FPR 10187991 IC50 = 160 nM T09960 CXK43P 10204589 IC50 = 3200 nM T09960 C4OM2Z 10205915 IC50 = 3000 nM T09960 CWC7X1 10208080 IC50 = 11 nM T09960 CS27UD 10208679 IC50 = 68 nM T09960 CO2T6R 10228759 IC50 = 50 nM T09960 C72HMR 10228761 IC50 = 17 nM T09960 CE95ZB 10230510 IC50 = 229000 nM T09960 CK49NQ 10272003 IC50 = 2900 nM T09960 C3CZ7H 10277466 IC50 = 20 nM T09960 CM6SE7 10280445 IC50 = 1 nM T09960 CE9ID0 10280944 IC50 = 6.1 nM T09960 C80DZB 10290194 IC50 = 89 nM T09960 CO0P4F 10301330 IC50 = 94 nM T09960 CWFB30 10323427 IC50 > 1000 nM T09960 CFAU91 10325578 IC50 = 7 nM T09960 CRZD69 10347790 IC50 = 0.2999 nM T09960 CQP8C4 10348408 IC50 = 5 nM T09960 CPU68L 10369469 IC50 = 0.3 nM T09960 CU5F2P 10371054 IC50 = 3981.07 nM T09960 C2Y8DC 10393635 IC50 = 1023.29 nM T09960 CV60SK 10413034 IC50 = 0.9 nM T09960 CYXB38 10414981 IC50 = 0.2 nM T09960 CJ6X4K 10416552 IC50 = 20417.38 nM T09960 CZK8R4 10425374 IC50 = 154000 nM T09960 CME0U1 10438399 IC50 = 3 nM T09960 CL75IC 10445499 IC50 = 20000 nM T09960 CFD3H2 10461319 IC50 = 7 nM T09960 CI3X4T 10462202 IC50 = 1.5 nM T09960 C2D5KO 10483364 IC50 = 141.25 nM T09960 CS8A6G 10531271 IC50 = 1100 nM T09960 C2YBW0 10555236 IC50 = 660 nM T09960 C96PZF 10617034 Ki = 2 nM T09960 C2N8IQ 10627515 IC50 = 110 nM T09960 C45TVD 10648217 IC50 = 840 nM T09960 C62DKM 10650855 IC50 = 380 nM T09960 CNV4E6 10695549 IC50 = 3200 nM T09960 CT9Y3K 10698789 IC50 = 6.8 nM T09960 C1TZO6 10746493 IC50 = 1.4 nM T09960 CDLS35 10746690 IC50 = 3.1 nM T09960 CRY4I7 10747204 IC50 = 2.2 nM T09960 CCG8V9 10792796 IC50 = 570 nM T09960 C87XAH 10793079 IC50 = 1200 nM T09960 CSWN32 10840407 IC50 = 430 nM T09960 C8W7IY 10840676 IC50 = 620 nM T09960 C5XMK1 10840679 IC50 = 390 nM T09960 CJK35A 10841420 IC50 = 3.3 nM T09960 CCDO97 10842229 IC50 = 3.8 nM T09960 CW9A7C 11069824 Ki = 275 nM T09960 C15AOC 11154101 IC50 = 4700 nM T09960 CVB54S 11157818 IC50 = 60 nM T09960 C2MFC7 11166533 IC50 = 449.78 nM T09960 C7V6JL 11177360 IC50 = 149.97 nM T09960 C6FK0H 11180743 IC50 = 30 nM T09960 CI05VQ 11189082 IC50 = 49 nM T09960 C8M4RU 11192476 IC50 = 34 nM T09960 CXF20N 11193076 IC50 = 130 nM T09960 CPRH05 11204141 IC50 = 60 nM T09960 CD98SL 11204472 IC50 = 1050 nM T09960 CKO02A 11210440 IC50 = 599.79 nM T09960 C2RBU8 11215601 IC50 = 50 nM T09960 CIS29O 11215950 IC50 = 89 nM T09960 CZ20TE 11224188 IC50 = 10100 nM T09960 CA39QR 11227406 IC50 > 1000 nM T09960 CN84TM 11234566 IC50 = 40000 nM T09960 CN51JH 11238728 IC50 = 50 nM T09960 C21OTD 11246827 IC50 = 149.97 nM T09960 CAR46F 11249997 IC50 = 4800 nM T09960 CS9I8P 11250534 IC50 = 70 nM T09960 CA5ST9 11259200 IC50 = 8500 nM T09960 C31MVR 11261876 IC50 = 40 nM T09960 CQ6KW0 11272103 IC50 = 1000 nM T09960 C06TUD 11285791 IC50 = 0.1 nM T09960 C5DG8M 11326950 IC50 = 349.95 nM T09960 C1A5ET 11329244 IC50 = 1000 nM T09960 CI3YG0 11342750 IC50 = 68 nM T09960 C5LK1F 11342841 IC50 = 25 nM T09960 C74ZPM 11350639 IC50 = 1400 nM T09960 CSAD06 11353001 IC50 = 1.1 nM T09960 CCZN17 11365412 IC50 = 40 nM T09960 CBZ18L 11376667 IC50 = 50 nM T09960 C8DJL6 11399408 IC50 = 30 nM T09960 C6RQ0D 11408704 IC50 = 1300 nM T09960 C5UZ6O 11410758 IC50 = 130 nM T09960 C7T9JS 11421221 IC50 = 13 nM T09960 C19RCV 11422270 IC50 = 30 nM T09960 C1E6KF 11433338 IC50 = 26 nM T09960 C6VCP5 11433740 IC50 = 30 nM T09960 CBEF39 11444710 IC50 = 140 nM T09960 CS6LA7 11466794 IC50 = 19 nM T09960 C7Z9KU 11467704 IC50 = 1.995 nM T09960 C6ZI2E 11478988 IC50 = 40 nM T09960 CW6YN0 11490468 IC50 = 140 nM T09960 C40IMW 11502371 IC50 = 1000 nM T09960 CA3SW7 11503459 IC50 = 2 nM T09960 CGN4S8 11505350 IC50 = 1.7 nM T09960 C3LBY6 11513274 IC50 = 0.21 nM T09960 C8P4GL 11520480 IC50 = 25 nM T09960 C4XVL8 11520510 IC50 = 67 nM T09960 CYH8J9 11525100 IC50 = 1.2 nM T09960 C7HF1B 11527582 IC50 = 12 nM T09960 C7LP9F 11527691 IC50 = 4.7 nM T09960 C0F7SR 11534473 IC50 = 1610 nM T09960 C0NL5U 11569805 IC50 = 84 nM T09960 CLY5O2 11570431 IC50 = 220 nM T09960 CE5KD2 11570778 IC50 = 2.8 nM T09960 C70EYD 11577846 IC50 = 3.2 nM T09960 C4KQI5 11578088 IC50 = 730 nM T09960 CAS56U 11585418 IC50 = 3.9 nM T09960 CEC49G 11585625 IC50 = 4.1 nM T09960 C1DKF4 11598797 IC50 = 610 nM T09960 CJ1IF0 11605997 IC50 = 1.2 nM T09960 C84YPR 11606411 IC50 = 630 nM T09960 C7C8FX 11626984 IC50 = 9 nM T09960 C57RHQ 11634966 IC50 = 860 nM T09960 C9CKA0 11635721 IC50 = 1.7 nM T09960 C54OFG 11636141 IC50 = 0.95 nM T09960 CJ3I2L 11639993 IC50 > 1000 nM T09960 CZ1T4W 11641131 IC50 = 8 nM T09960 C0XZK5 11650548 IC50 = 0.19 nM T09960 CH97IX 11656080 IC50 = 21.5 nM T09960 CU7OG2 11669935 IC50 = 283 nM T09960 CFV0I9 11690481 IC50 = 17 nM T09960 CPIY98 11692945 IC50 = 6.4 nM T09960 C6WD8L 11693007 IC50 = 20 nM T09960 C17RPK 11700429 IC50 = 0.48 nM T09960 CCG50D 11753754 IC50 = 190 nM T09960 CHS9Q3 11785237 IC50 < 0.1 nM T09960 CFA15U 11786927 IC50 = 10 nM T09960 C9OTN2 11787124 IC50 = 76 nM T09960 C2J8RH 11844212 IC50 = 30 nM T09960 CL1FX0 11947758 IC50 = 380.19 nM T09960 CGP04N 11988311 IC50 = 0.137 nM T09960 CJX31Q 12093170 IC50 = 703 nM T09960 CK80NA 12987698 EC50 = 1900 nM T09960 CJGC50 14434082 EC50 = 10000 nM T09960 C8L9VX 15485365 IC50 = 1000 nM T09960 CIZ8C1 15783796 EC50 = 1995.26 nM T09960 CCDX50 15940498 IC50 = 0.5 nM T09960 CU02IX 15940799 IC50 = 0.3 nM T09960 CN4F8X 15940800 IC50 = 0.1 nM T09960 C8JIP7 15940801 IC50 = 0.4 nM T09960 CTH2A9 15941083 IC50 = 0.4 nM T09960 CF30UM 15941086 IC50 = 0.1 nM T09960 CM10PF 15941255 IC50 = 0.08 nM T09960 C5WUJ0 15942352 IC50 = 48.4 nM T09960 CB8H6M 15947119 IC50 = 0.2 nM T09960 C3UW0T 15950679 IC50 = 18.9 nM T09960 C2U1GH 15958353 IC50 = 20 nM T09960 CCL59Z 16007088 IC50 = 0.32 nM T09960 CXBD17 16041224 IC50 = 6.6 nM T09960 CDU1L0 16041411 IC50 = 0.9 nM T09960 CGM4N8 16041594 IC50 = 15.7 nM T09960 CYA3K5 16064151 IC50 = 10 nM T09960 C38DNF 16073659 IC50 = 780 nM T09960 CZ5JG1 16073660 IC50 = 0.76 nM T09960 CQI01L 16073661 IC50 = 46 nM T09960 CS48RO 16073662 IC50 = 1 nM T09960 C71ODK 16073663 IC50 = 21 nM T09960 C05TIF 16073664 IC50 = 132 nM T09960 C36HRZ 16073665 IC50 = 20 nM T09960 C74ROH 16073666 IC50 = 25 nM T09960 CAK3O1 16073667 IC50 = 20 nM T09960 CO0J6E 16073668 IC50 = 560 nM T09960 C63SFG 16073669 IC50 = 32 nM T09960 CLM4I9 16073670 IC50 = 1.1 nM T09960 C3W6XJ 16073671 IC50 = 500 nM T09960 C3P8HL 16073672 IC50 = 110 nM T09960 CIWA92 16073673 IC50 = 56 nM T09960 C3Y0MT 16073674 IC50 = 25 nM T09960 C9G8TZ 16124598 IC50 = 251.19 nM T09960 CI32YP 16301115 EC50 = 13500 nM T09960 CUTB83 16655051 IC50 = 92.9 nM T09960 C3WX9K 16658855 IC50 = 6530 nM T09960 C7X0TS 16659334 IC50 = 3.5 nM T09960 CG7MA3 16726107 EC50 = 1100 nM T09960 CM0QJ2 16728324 IC50 = 8.75 nM T09960 CIFJ10 16728325 IC50 = 6.22 nM T09960 C3TNU9 16728326 IC50 = 122 nM T09960 C8UMZ1 16728609 IC50 = 599.79 nM T09960 C2YBX3 16728610 IC50 = 1900 nM T09960 C49PQF 16728611 IC50 = 800 nM T09960 CV9ZH3 16728612 IC50 = 600 nM T09960 CZ9TG7 16728613 IC50 = 480 nM T09960 C9CKU7 16728614 IC50 = 1999.86 nM T09960 CZV0H1 16728615 IC50 = 899.5 nM T09960 CGSC15 16728616 IC50 = 1698.24 nM T09960 CV54TY 16728617 IC50 = 5700 nM T09960 CJ1YK4 16728618 IC50 = 1300 nM T09960 CIM1Z9 16728619 IC50 = 1599.56 nM T09960 CY97UR 16728620 IC50 = 39000 nM T09960 C8H9RN 16728621 IC50 = 500.03 nM T09960 CUC7B5 16728622 IC50 = 1698.24 nM T09960 CED81G 16728623 IC50 = 699.84 nM T09960 CB45LR 16728624 IC50 = 2897.34 nM T09960 C9BHE4 16728625 IC50 = 1698.24 nM T09960 C8X7LT 16728626 IC50 = 1100 nM T09960 C6KDW9 16728627 IC50 = 3700 nM T09960 C3UN0X 16728628 IC50 = 8700 nM T09960 CHBQ91 16728629 IC50 = 600 nM T09960 C58IKH 16728630 IC50 = 1199.5 nM T09960 CE51NB 16728631 IC50 = 3404.08 nM T09960 C7JDU0 16728632 IC50 = 3100 nM T09960 CMG1V0 16728633 IC50 > 30000 nM T09960 C1W2VH 16728634 IC50 > 30000 nM T09960 CHQO72 16728635 IC50 = 600 nM T09960 CT7G2R 16728636 IC50 > 30000 nM T09960 CW10DK 16728637 IC50 > 30000 nM T09960 CUP1Q0 16728638 IC50 > 30000 nM T09960 C4EG0L 16728639 IC50 > 30000 nM T09960 CQP2C6 16728640 IC50 > 30000 nM T09960 CWK46L 16728641 IC50 > 30000 nM T09960 C2V1FK 16728642 IC50 = 8500 nM T09960 CD8U4Z 16728643 IC50 = 139.96 nM T09960 CS9FH8 16728644 IC50 = 399.94 nM T09960 C6LWX7 16728645 IC50 = 4197.59 nM T09960 CZU94T 16728646 IC50 > 30000 nM T09960 CD6AM7 16728647 IC50 = 749.89 nM T09960 C0CU2F 16728648 IC50 = 14000 nM T09960 CL9N1W 16728649 IC50 = 1999.86 nM T09960 C0E3SL 16728783 IC50 > 3000 nM T09960 CS1F3B 16728784 IC50 = 28 nM T09960 CFCV60 16728785 IC50 = 130 nM T09960 CDMA29 16728786 IC50 = 53 nM T09960 CAX2B7 16728787 IC50 = 1.1 nM T09960 CQ7G2U 16728788 EC50 = 2000 nM T09960 C9H8IS 16730521 IC50 = 11 nM T09960 CP4CY0 18442936 IC50 = 37 nM T09960 CTM71O 20664115 IC50 = 12 nM T09960 CES60Q 20664141 IC50 = 7 nM T09960 CB36XZ 20664149 IC50 = 0.8 nM T09960 CXOS35 20664156 IC50 = 2.5 nM T09960 C7RO9I 20664159 IC50 = 8.2 nM T09960 C87RFX 20664160 IC50 = 65 nM T09960 CFQM24 20664161 IC50 = 0.42 nM T09960 CUZ8P0 20664163 IC50 = 2.799 nM T09960 CBJ5N8 20672360 IC50 = 0.5 nM T09960 CLE46M 20672362 IC50 = 0.3 nM T09960 CS20IY 20672370 IC50 = 0.3 nM T09960 CJXP29 20672384 IC50 = 0.84 nM T09960 C2DEH4 20672386 IC50 = 0.5 nM T09960 C2PG9O 21064126 IC50 = 79 nM T09960 CFWJ06 21064281 IC50 = 28 nM T09960 CHC4Q3 21064283 IC50 = 13 nM T09960 CS78PF 21064289 IC50 = 92 nM T09960 C3K0IQ 21064293 IC50 = 130 nM T09960 CDU03R 21064295 IC50 = 33 nM T09960 C5R4DC 21064297 IC50 = 79 nM T09960 CND40Q 21064299 IC50 = 40 nM T09960 CS6IT0 21064329 IC50 = 86 nM T09960 CTMC32 21064331 IC50 = 170 nM T09960 CA1E0H 21064338 IC50 = 450 nM T09960 C8NTA6 21147749 IC50 = 2 nM T09960 CY0J1U 21148035 IC50 = 1000 nM T09960 CE38ZB 21341080 IC50 = 1.6 nM T09960 C9YZ3A 21867666 IC50 = 7 nM T09960 CKGT37 21925890 IC50 = 570 nM T09960 CE05FA 21926122 IC50 > 3000 nM T09960 C4WX7Q 21926246 IC50 > 3000 nM T09960 C0UT7V 21926618 IC50 = 69 nM T09960 CWH1D9 21926948 IC50 = 52 nM T09960 C3E0DK 21927225 IC50 = 54 nM T09960 CE2P5B 21927257 IC50 = 590 nM T09960 CO9VD3 22135856 IC50 > 3000 nM T09960 C8HE4I 23285265 IC50 = 720 nM T09960 CXF8Z9 23294208 IC50 = 19952.62 nM T09960 C3XN1D 23294214 IC50 = 1584.89 nM T09960 C32CYE 23577328 IC50 = 33000 nM T09960 CQ4M2S 23577360 IC50 = 39000 nM T09960 C1VX7E 23577362 IC50 = 3500 nM T09960 C6P2HL 23577370 IC50 = 2800 nM T09960 C5ZSO4 23577378 IC50 = 7100 nM T09960 CAX0O6 23577382 IC50 = 7400 nM T09960 C3U9PK 23577386 IC50 = 1400 nM T09960 C7SD8Q 23577388 IC50 = 34000 nM T09960 C16ZJO 23577409 IC50 = 13000 nM T09960 C6SB3P 23577448 IC50 = 30000 nM T09960 CP2RA0 23577500 IC50 > 3000 nM T09960 CE29IW 23650547 IC50 = 1 nM T09960 C7JV4W 23725177 IC50 = 780 nM T09960 C25HKJ 24758044 IC50 > 20000 nM T09960 C4AEG2 25024699 IC50 = 1.7 nM T09960 C5M2CK 25057602 IC50 = 144 nM T09960 C91NVS 25057877 IC50 = 300 nM T09960 C6MO8Z 25130569 IC50 = 3467.37 nM T09960 CUH0C9 25130571 IC50 = 9332.54 nM T09960 C4MR8V 25130901 IC50 = 776.25 nM T09960 CE30DM 25130903 IC50 = 5248.07 nM T09960 CO4VZ3 25130904 IC50 > 31622.78 nM T09960 C4OY2V 25131220 IC50 > 31622.78 nM T09960 C0J1OY 25131899 IC50 > 31622.78 nM T09960 C3N2LV 25131900 IC50 = 19952.62 nM T09960 CCPA34 25131901 IC50 = 1258.93 nM T09960 CJG1U8 25131902 IC50 = 3981.07 nM T09960 CWA93M 25132253 IC50 = 63.1 nM T09960 C3I1XJ 25132254 IC50 = 5.012 nM T09960 CY52ZQ 25132255 IC50 = 19.95 nM T09960 CM30EC 25132603 IC50 = 1 nM T09960 CK0L3W 25132604 IC50 = 5.012 nM T09960 C4GF3T 25132945 IC50 = 2398.83 nM T09960 C1WAP7 25132946 IC50 = 9332.54 nM T09960 CY8R6L 25132948 IC50 > 31622.78 nM T09960 COK24W 25133270 IC50 = 7079.46 nM T09960 CGR54C 25133271 IC50 = 446.68 nM T09960 CTQ2C7 25133617 IC50 = 5011.87 nM T09960 C8R5JI 25133618 IC50 = 7943.28 nM T09960 C28FCZ 25133619 IC50 = 8511.38 nM T09960 C9PCN5 25133620 IC50 = 4570.88 nM T09960 CQ4ZJ9 25133961 IC50 = 63.1 nM T09960 C0XNZ7 25133962 IC50 = 15.85 nM T09960 CIY4Q3 25133963 IC50 = 5.248 nM T09960 C2LZN5 25133964 IC50 = 29.51 nM T09960 C54KPB 25205600 IC50 = 65 nM T09960 C6J3TG 25205601 IC50 = 84 nM T09960 CE0WO1 25205764 IC50 = 43 nM T09960 CR49UP 25205766 IC50 = 20 nM T09960 CV02HS 25205767 IC50 = 12 nM T09960 CBH92X 25205921 IC50 = 27 nM T09960 C84EQC 25205923 IC50 = 6 nM T09960 CH4ZW0 25206069 IC50 = 90 nM T09960 CW0FH8 25206070 IC50 = 21 nM T09960 C6HWA7 25206071 IC50 = 26 nM T09960 C2K9DX 25206204 IC50 = 60 nM T09960 C13FTZ 25206227 IC50 = 34 nM T09960 C0VWM1 25206397 IC50 = 32 nM T09960 C2GU6Q 25230769 IC50 > 500 nM T09960 C7SUF3 25230770 IC50 = 217 nM T09960 CQP83X 25230771 IC50 = 19 nM T09960 CRCS05 25230773 IC50 = 19 nM T09960 CO9T8A 25230826 IC50 = 18 nM T09960 C8WF3A 25230827 IC50 = 22 nM T09960 C54LQF 25230828 IC50 = 30 nM T09960 CR31QN 25230829 IC50 = 25 nM T09960 C2M8SR 25230896 IC50 = 349 nM T09960 CT21IO 25230897 IC50 = 60 nM T09960 CB9V4X 25230898 IC50 = 22 nM T09960 CH6N1A 25230899 IC50 = 27 nM T09960 CKH70V 25230969 IC50 > 500 nM T09960 CVXD97 25230970 IC50 = 11 nM T09960 CU1W0E 25230971 IC50 = 80 nM T09960 CJ54KN 25231038 IC50 = 70 nM T09960 CV2L4K 25231041 IC50 = 64 nM T09960 COQI09 25231105 IC50 = 78 nM T09960 CBMH73 25256856 IC50 = 2 nM T09960 CJ0ZN4 25256857 IC50 = 8 nM T09960 C2FZ9P 42606792 IC50 = 1636 nM T09960 CI1C5U 42623163 IC50 = 2 nM T09960 C4HL1I 44129650 IC50 = 37.3 nM T09960 CEKX13 44194496 IC50 = 113.6 nM T09960 CV9M8D 44194587 IC50 = 3.32 nM T09960 C4AZ9G 44194588 IC50 = 1.53 nM T09960 C0Q5SE 44194589 IC50 = 2.1 nM T09960 CY0V2U 44194590 IC50 = 1.09 nM T09960 CM7OY9 44194675 IC50 = 5 nM T09960 C4BJA6 44194676 IC50 = 2.93 nM T09960 C1PT3U 44205000 IC50 = 0.9 nM T09960 C5YFB9 44252324 IC50 > 10000 nM T09960 CM67JX 44273531 IC50 = 0.1 nM T09960 CEF2O4 44273816 IC50 = 1.1 nM T09960 C7P5EI 44273830 IC50 = 0.2 nM T09960 COX48Y 44273846 IC50 = 1000 nM T09960 CJ4H3K 44273850 IC50 = 51 nM T09960 CY31BC 44273872 IC50 = 1.5 nM T09960 C1G9IF 44273888 IC50 = 0.4 nM T09960 CG46IJ 44273960 IC50 = 0.7998 nM T09960 CU5O9Q 44273996 IC50 = 0.4 nM T09960 CO8VE2 44274022 IC50 = 3.7 nM T09960 C7MZA3 44274042 IC50 = 4.797 nM T09960 CTB92I 44274043 IC50 = 0.2 nM T09960 CJOD81 44274090 IC50 = 1.6 nM T09960 CG8A6Y 44274106 IC50 = 0.9 nM T09960 CM4VI3 44274108 IC50 = 0.8 nM T09960 CW5KM0 44322729 IC50 = 70 nM T09960 CN3YT4 44324386 IC50 = 4000 nM T09960 CV1G7P 44325489 IC50 = 19 nM T09960 CY3L7S 44325511 IC50 = 220 nM T09960 CJC29B 44325542 IC50 = 4 nM T09960 C5BJ1O 44325665 IC50 = 0.8 nM T09960 CW36ZF 44325710 IC50 = 22 nM T09960 C47CDP 44325917 IC50 = 22 nM T09960 CTL92Q 44332341 IC50 = 0.2 nM T09960 C7SNJ5 44332489 IC50 = 0.4 nM T09960 C03NLX 44332684 IC50 = 0.1 nM T09960 CQT3M4 44332814 IC50 = 1 nM T09960 CJQA92 44335765 IC50 = 10 nM T09960 C2TEM7 44336415 IC50 = 20 nM T09960 CPGN89 44337326 Ki = 1 nM T09960 C5OE3P 44341106 Ki = 2 nM T09960 C0K5BM 44342961 IC50 = 0.23 nM T09960 CED6Z5 44342962 IC50 = 0.23 nM T09960 C8ON9S 44356876 IC50 = 21 nM T09960 C60YTZ 44356944 IC50 = 1.5 nM T09960 CHN56D 44356952 IC50 = 1.2 nM T09960 CBFY26 44357063 IC50 = 1.2 nM T09960 CSL5R9 44357072 IC50 = 0.8 nM T09960 CHM12S 44357078 IC50 = 0.5 nM T09960 C64KXD 44357079 IC50 = 0.4 nM T09960 CK9G2U 44357375 IC50 = 1.7 nM T09960 C7CMB3 44357379 IC50 = 1.1 nM T09960 CZTI85 44373672 IC50 = 27 nM T09960 C48ELJ 44373721 IC50 = 5 nM T09960 CDP34B 44373748 IC50 = 86 nM T09960 CZU19Q 44373755 IC50 ~ 27 nM T09960 CWM1F5 44373756 IC50 = 0.13 nM T09960 CJ6X0R 44373767 IC50 = 69 nM T09960 C5F3AQ 44373768 IC50 = 33 nM T09960 C0I1AL 44373852 IC50 = 5 nM T09960 C4QN7Z 44373926 IC50 = 6 nM T09960 CD64UI 44373973 IC50 = 14 nM T09960 C4ZCA2 44374016 IC50 = 8 nM T09960 CHD26R 44374017 IC50 = 43 nM T09960 CG14HU 44374086 IC50 = 30 nM T09960 C4B8ZF 44374088 IC50 = 11 nM T09960 COT83J 44374136 IC50 = 46 nM T09960 C76UBK 44383760 IC50 = 41 nM T09960 C60VEP 44383787 IC50 = 2.1 nM T09960 C74DCF 44384011 IC50 = 11.5 nM T09960 C09IYH 44384012 IC50 = 23 nM T09960 C4A3GF 44384584 IC50 = 1 nM T09960 CCK72Y 44384642 IC50 = 4.4 nM T09960 CE0S9Q 44384705 IC50 = 6.9 nM T09960 CG9K8P 44384782 IC50 = 0.5 nM T09960 CH6J3Q 44384875 IC50 = 1.2 nM T09960 CO9P8X 44384927 IC50 = 0.8 nM T09960 C3QL8D 44384969 IC50 = 11 nM T09960 CUCH65 44385583 IC50 = 0.5 nM T09960 CQ58FI 44389412 IC50 = 3.6 nM T09960 C4PH3E 44392074 IC50 = 91 nM T09960 C8UZX0 44392078 IC50 = 8700 nM T09960 CHMY61 44392082 IC50 = 3600 nM T09960 CDN01K 44392083 IC50 = 3500 nM T09960 CWJK96 44392084 IC50 = 690 nM T09960 C2VN8S 44392087 IC50 < 10 nM T09960 CN0H4K 44392088 IC50 = 46 nM T09960 C8B9XD 44392092 IC50 = 2200 nM T09960 CM5F6G 44392093 IC50 = 2300 nM T09960 C3E6SV 44392094 IC50 = 180 nM T09960 CWY84B 44392095 IC50 = 7900 nM T09960 C27ISR 44392096 IC50 = 76 nM T09960 C91WEC 44392103 IC50 = 630 nM T09960 CC8L5E 44392104 IC50 = 4900 nM T09960 CR5NG8 44392105 IC50 = 800 nM T09960 C98EUH 44392106 IC50 = 370 nM T09960 C98COA 44392109 IC50 = 5500 nM T09960 CZ1A4U 44392110 IC50 = 580 nM T09960 C4CHI6 44392111 IC50 = 110 nM T09960 CH90MX 44392114 IC50 = 470 nM T09960 CT3V8A 44392115 IC50 = 5900 nM T09960 CXU52S 44392116 IC50 = 780 nM T09960 C7MIY0 44392117 IC50 = 290 nM T09960 CI5S1Q 44392123 IC50 = 770 nM T09960 CQ3UK0 44392124 IC50 = 650 nM T09960 CIHT56 44392125 IC50 = 33 nM T09960 CAS85F 44392126 IC50 = 4100 nM T09960 C2G1OP 44392130 IC50 = 150 nM T09960 C4F9EW 44392131 IC50 = 2100 nM T09960 CN3B8U 44392132 IC50 = 2600 nM T09960 C9O8VP 44392135 IC50 = 5900 nM T09960 CX69VZ 44392136 IC50 = 2700 nM T09960 CXO91S 44392137 IC50 = 32 nM T09960 C6X1LF 44392142 IC50 = 310 nM T09960 CZOV60 44392143 IC50 = 370 nM T09960 CM83HG 44392144 IC50 = 1900 nM T09960 C4H0PT 44392147 IC50 = 1100 nM T09960 C3PHL1 44392148 IC50 = 680 nM T09960 CK27GP 44392149 IC50 = 310 nM T09960 C7KXJ0 44392153 IC50 = 66 nM T09960 CMZ6P9 44392154 IC50 = 7200 nM T09960 CGU0F6 44392155 IC50 = 1400 nM T09960 CCTR59 44392159 IC50 = 190 nM T09960 C3TCB0 44392160 IC50 = 6800 nM T09960 CXZU54 44392161 IC50 = 60 nM T09960 C0MN1I 44392162 IC50 = 350 nM T09960 C72VXL 44392166 IC50 = 580 nM T09960 CR4JP7 44392167 IC50 = 38 nM T09960 C31FMI 44392168 IC50 = 5100 nM T09960 CXUA20 44392169 IC50 = 660 nM T09960 CQTD48 44392176 IC50 = 49 nM T09960 CJ4QA3 44392196 IC50 = 240 nM T09960 C3QNW5 44392203 IC50 = 680 nM T09960 C70TGZ 44392204 IC50 = 560 nM T09960 C9BM2F 44392211 IC50 = 1800 nM T09960 CQWI02 44392213 IC50 = 320 nM T09960 CY5TX7 44392218 IC50 = 7400 nM T09960 CV41WR 44392219 IC50 = 3400 nM T09960 CMVR86 44392220 IC50 = 110 nM T09960 CAZ5I4 44392229 IC50 = 100 nM T09960 CSNB94 44392235 IC50 = 35 nM T09960 CHU5K6 44392244 IC50 = 62 nM T09960 CBA56P 44392253 IC50 = 42 nM T09960 CHT1S5 44392258 IC50 = 5400 nM T09960 CO5D7H 44395365 IC50 = 7200 nM T09960 CEY49R 44395386 IC50 = 8800 nM T09960 C0ZFD8 44401488 IC50 = 0.35 nM T09960 CHQY70 44401593 IC50 = 63 nM T09960 CL24ST 44401608 IC50 = 200 nM T09960 CQC16I 44401686 IC50 = 2.6 nM T09960 CFR53O 44401731 IC50 = 10 nM T09960 CEKA14 44401734 IC50 = 100 nM T09960 CATD12 44401751 IC50 = 0.89 nM T09960 C16MBG 44401760 IC50 = 0.82 nM T09960 CWH26M 44401763 IC50 = 12 nM T09960 CD3X4N 44401765 IC50 = 6.3 nM T09960 CH65CZ 44401863 IC50 = 12 nM T09960 CT9XO0 44401956 IC50 = 0.5 nM T09960 CJ9FS4 44401965 IC50 = 0.6 nM T09960 C8WV0Q 44401985 IC50 = 23 nM T09960 CQ6SO2 44404596 IC50 = 8.5 nM T09960 C15PRG 44404601 IC50 = 760 nM T09960 CA15WI 44404605 IC50 = 310 nM T09960 CL86FA 44404638 IC50 = 200 nM T09960 CTM2X0 44404639 IC50 = 26 nM T09960 C98QDP 44404640 IC50 = 5.9 nM T09960 CGD3Z5 44404641 IC50 = 130 nM T09960 CTC28Z 44404642 IC50 = 22 nM T09960 C34CQF 44404643 IC50 = 24 nM T09960 CVK07T 44404644 IC50 = 11 nM T09960 CMCP98 44404645 IC50 = 740 nM T09960 CZI0D9 44404650 IC50 = 19 nM T09960 CSY85U 44404656 IC50 = 105 nM T09960 CO28NW 44404657 IC50 = 7.9 nM T09960 C0J5YT 44404658 IC50 = 9.1 nM T09960 CE0CM4 44404692 IC50 = 58 nM T09960 CN30IB 44404697 IC50 = 78 nM T09960 CTFY36 44404702 IC50 = 28 nM T09960 C1CBI7 44404705 IC50 = 2.3 nM T09960 CM50EI 44404709 IC50 = 7.1 nM T09960 C5VJ9P 44404710 IC50 = 260 nM T09960 C6RAG1 44404716 IC50 < 1 nM T09960 CH3NG1 44404719 IC50 = 6.3 nM T09960 C01ZEW 44404720 IC50 = 85 nM T09960 CU9BI1 44404724 IC50 = 12 nM T09960 CD3X0F 44404730 IC50 = 200 nM T09960 CV9YH2 44412984 IC50 = 40 nM T09960 C4LT3K 44415740 IC50 = 20 nM T09960 C5U1EA 44415755 IC50 = 0.7 nM T09960 CUG6N2 44415756 IC50 = 250 nM T09960 CHU9Y6 44415783 IC50 = 70 nM T09960 C1NGI4 44415784 IC50 = 50 nM T09960 C9GO0B 44415800 IC50 = 2 nM T09960 C64VRB 44415820 IC50 = 6 nM T09960 CRJ70D 44415821 IC50 = 39 nM T09960 CT73JO 44415847 IC50 = 5 nM T09960 CMA02E 44431926 IC50 = 1300 nM T09960 CTO19K 44431931 IC50 > 30000 nM T09960 C4RST8 44431934 IC50 > 30000 nM T09960 CZ4YP3 44431944 IC50 = 279.9 nM T09960 CVMN01 44431946 IC50 = 3097.42 nM T09960 CHL9M6 44431949 IC50 = 389.94 nM T09960 CXY1F8 44431951 IC50 = 400 nM T09960 CK65WG 44431953 IC50 = 1300 nM T09960 C3E5DV 44431954 IC50 = 349.95 nM T09960 CV5CN0 44431959 IC50 = 579.43 nM T09960 C3UJ8R 44431962 IC50 = 579.43 nM T09960 C60EHY 44431965 IC50 = 1099.01 nM T09960 C7OVB6 44431967 IC50 = 210 nM T09960 C40LUV 44431969 IC50 = 1500 nM T09960 CG2AB4 44431971 IC50 = 320 nM T09960 C2SVT3 44431972 IC50 = 57 nM T09960 CQED73 44431975 IC50 = 450 nM T09960 C9JM4F 44431976 IC50 = 170 nM T09960 C80MVI 44431977 IC50 = 100 nM T09960 C7P2RW 44431979 IC50 = 47 nM T09960 C8XTN1 44431984 IC50 = 35 nM T09960 CHK5S9 44431986 IC50 = 27 nM T09960 CT93GC 44439155 IC50 = 63 nM T09960 CJPR21 44439313 IC50 = 93 nM T09960 CXU41O 44439314 IC50 = 400 nM T09960 CDFP30 44447731 IC50 = 2 nM T09960 CFAL15 44447732 IC50 = 1.3 nM T09960 C9EM8Q 44447733 IC50 = 6.5 nM T09960 CX89DC 44447734 IC50 = 0.8 nM T09960 CHKC89 44447735 IC50 = 1.8 nM T09960 CWB20Y 44454972 IC50 = 48 nM T09960 C4KX7W 44454975 IC50 = 539 nM T09960 CJZ7N1 44454977 IC50 = 4 nM T09960 C6RQY0 44454999 IC50 = 15 nM T09960 C06XYR 44455001 IC50 = 100 nM T09960 C2G0ZQ 44455031 IC50 = 27 nM T09960 CD12BW 44455033 IC50 = 53 nM T09960 C3FE8U 44455034 IC50 = 381 nM T09960 C4TFR9 44455069 IC50 = 4 nM T09960 CMF34Z 44455072 IC50 = 29 nM T09960 C3BVO1 44455103 IC50 = 271 nM T09960 CTU7H3 44455106 IC50 = 323 nM T09960 CY40FE 44455143 IC50 = 96 nM T09960 CW96PA 44455144 IC50 = 20 nM T09960 CNZ60R 44455177 IC50 = 271 nM T09960 C70PHB 44455180 IC50 = 78 nM T09960 CL12VU 44455217 IC50 = 0.4 nM T09960 C7KS8J 44455223 IC50 = 31 nM T09960 C7C1PI 44455225 IC50 = 310 nM T09960 CCA13O 44455313 IC50 = 970 nM T09960 CHEP83 44461014 IC50 > 10000 nM T09960 CME3S8 44461016 IC50 > 10000 nM T09960 CUX8D6 44461274 IC50 = 6 nM T09960 C7LQY9 44461275 IC50 = 3 nM T09960 CY32GT 44461476 IC50 = 5 nM T09960 C8JY5Z 44461494 IC50 = 35 nM T09960 CL5AM7 44461513 IC50 = 40 nM T09960 C31UNS 44461521 IC50 = 15 nM T09960 CE62UH 44461522 IC50 = 20 nM T09960 C3OTS5 44461559 IC50 = 15 nM T09960 COQZ58 44461560 IC50 = 100 nM T09960 CVC83W 44461561 IC50 = 25 nM T09960 CRZ8B2 44461581 IC50 = 39.81 nM T09960 CZH18E 44461603 IC50 = 35 nM T09960 C7PD1X 44461623 IC50 = 120 nM T09960 C2VW8I 44461628 IC50 = 10 nM T09960 CQ5XM0 44461677 IC50 = 5 nM T09960 CHC7O1 44461684 IC50 = 2 nM T09960 C3KMA9 44461689 IC50 = 4 nM T09960 CR8L1S 44461699 IC50 = 3 nM T09960 CXHT47 44461707 IC50 = 2 nM T09960 CD2KC6 44461713 IC50 = 6 nM T09960 CREY18 44461714 IC50 = 10 nM T09960 CT78IZ 44461741 IC50 = 0.75 nM T09960 CSR9Q6 44461774 IC50 = 150 nM T09960 C30PZS 44461785 IC50 = 1000 nM T09960 C5MR0E 44461790 IC50 = 1000 nM T09960 C49OIF 44461804 IC50 = 794.33 nM T09960 CZ7IX1 44461817 IC50 = 3 nM T09960 CO9RF0 44461823 IC50 = 4 nM T09960 C3XIJ9 44461831 IC50 = 100 nM T09960 CG65UL 44461835 IC50 = 20 nM T09960 C3KJP5 44511861 IC50 = 40 nM T09960 C4N5ET 44511871 IC50 = 0.8 nM T09960 C3M8UD 44511934 IC50 = 0.3 nM T09960 C2ZFD8 44511935 IC50 = 0.6 nM T09960 COK7H1 44511938 IC50 = 0.3 nM T09960 CY9FT7 44511966 IC50 = 7 nM T09960 CHV3I6 44511967 IC50 = 10.9 nM T09960 CBSD16 44512001 IC50 = 0.7 nM T09960 CM85OE 44512058 IC50 = 0.3 nM T09960 CI4S8C 44512090 IC50 = 0.3 nM T09960 C6WH8N 44512349 IC50 = 1.3 nM T09960 CGM39D 44532866 IC50 = 265 nM T09960 CT5N4E 44555481 IC50 = 4 nM T09960 C7WO5E 44555482 IC50 = 27 nM T09960 CT8S2U 44559501 IC50 = 60000 nM T09960 CF1C8U 44564835 IC50 = 89.2 nM T09960 CL4N5D 44564884 IC50 = 85.3 nM T09960 C6P8OF 44564885 IC50 = 52.8 nM T09960 CK49AW 44564886 IC50 = 3.16 nM T09960 C8URX2 44564887 IC50 = 3.11 nM T09960 CA96BX 44564929 IC50 = 3.93 nM T09960 CJ0C6T 44564930 IC50 = 0.513 nM T09960 C5AVF0 44564931 IC50 = 164 nM T09960 C5U0TR 44564982 IC50 = 4.87 nM T09960 C8GCQ6 44564983 IC50 = 6.12 nM T09960 CE1OG0 44564984 IC50 = 28.7 nM T09960 CM4Z0V 44564985 IC50 = 315 nM T09960 C9JI2F 44565035 IC50 = 176 nM T09960 C37WSJ 44565036 IC50 = 187 nM T09960 CMOC65 44565037 IC50 = 0.84 nM T09960 CG2UO0 44565038 IC50 = 0.38 nM T09960 C3MNR0 44565080 IC50 = 0.48 nM T09960 CF6JG1 44565081 IC50 = 49.9 nM T09960 CA0FC1 44565082 IC50 = 1.3 nM T09960 C6DI0T 44565083 IC50 = 62 nM T09960 C8XF4D 44565557 IC50 = 3.499 nM T09960 CXT21C 44565558 IC50 = 28.97 nM T09960 C8BL9U 44565559 IC50 = 199.99 nM T09960 CXN35S 44565673 IC50 = 0.3999 nM T09960 C4ZMI3 44565674 IC50 = 3.6 nM T09960 CQ8CR4 44565718 IC50 = 0.8995 nM T09960 CUB24L 44565719 IC50 = 0.7998 nM T09960 CYK2S8 44565720 IC50 = 0.2999 nM T09960 CRN02H 44565721 IC50 = 3.7 nM T09960 C7IET0 44565742 IC50 = 0.5 nM T09960 CP4J3U 44565761 IC50 = 0.57 nM T09960 CKS65Z 44565762 IC50 = 0.5998 nM T09960 C3ZRO8 44565791 IC50 = 2.999 nM T09960 CIEU13 44565852 IC50 = 0.8892 nM T09960 C6R4PT 44565853 IC50 = 0.7603 nM T09960 CIS5B7 44565854 IC50 = 1 nM T09960 CYP76Z 44565874 IC50 = 13 nM T09960 CH0V8X 44568898 IC50 > 3162.28 nM T09960 CIZ10G 44570177 IC50 = 35 nM T09960 CZ65FC 44570267 IC50 = 19 nM T09960 CBHU64 44570268 IC50 = 37 nM T09960 CY5PT0 44570269 IC50 = 30 nM T09960 C8ZA1H 44570270 IC50 = 76 nM T09960 CFH4B9 44570307 IC50 = 104 nM T09960 C4XR6K 44573097 IC50 = 320 nM T09960 C9QV3T 44573098 IC50 = 129 nM T09960 CT2BF3 44573127 IC50 = 74 nM T09960 CSD69K 44573252 IC50 = 13 nM T09960 C24BDO 44573253 IC50 = 3 nM T09960 CP6S9W 44573254 IC50 = 4 nM T09960 C6V8OC 44573255 IC50 = 7 nM T09960 CA43WF 44573256 IC50 = 6 nM T09960 C3YHW1 44573297 IC50 = 21 nM T09960 C3P8EI 44573298 IC50 = 24 nM T09960 CS01PW 44573299 IC50 = 18 nM T09960 CC38YB 44573300 IC50 = 23 nM T09960 CL7KF4 44573301 IC50 = 13 nM T09960 C3H6AO 44573302 IC50 = 40 nM T09960 CS4AC6 44573335 IC50 = 11 nM T09960 CDI9P0 44573336 IC50 = 5 nM T09960 CA0P3K 44573337 IC50 = 7 nM T09960 CT9R5H 44573338 IC50 = 4 nM T09960 CQBA10 44573339 IC50 = 23 nM T09960 CH6Q4S 44573340 IC50 = 5 nM T09960 C03RHO 44573341 IC50 = 13 nM T09960 CIXC68 44590222 IC50 = 2490 nM T09960 CU71HW 44590230 IC50 = 37.5 nM T09960 C2HUS5 44590332 IC50 = 145 nM T09960 CGM7H6 44590394 IC50 = 1 nM T09960 CJ95XB 44590395 IC50 = 1230 nM T09960 CE5U9X 44590439 IC50 = 3 nM T09960 C81IGZ 44590440 IC50 = 0.5 nM T09960 C92IJZ 44590441 IC50 = 5800 nM T09960 CI1OX6 44590557 IC50 = 7.5 nM T09960 CS8ZR6 44590583 IC50 = 14 nM T09960 CR4K7Y 44590584 IC50 = 48 nM T09960 C6ZX0E 44590585 IC50 = 5 nM T09960 C4UR9F 44590586 IC50 = 0.05 nM T09960 CDR4P2 44590633 IC50 = 0.34 nM T09960 CWEQ65 44590634 IC50 = 0.48 nM T09960 CRE37W 44590635 IC50 = 0.94 nM T09960 CCBA38 44590681 IC50 = 0.07 nM T09960 C87MFS 44590682 IC50 = 1.54 nM T09960 C24KEF 44590683 IC50 = 2.33 nM T09960 C9QSX8 44590684 IC50 = 3.76 nM T09960 C9PC7J 44590704 IC50 = 24 nM T09960 CQ6SI3 44590717 IC50 = 13.4 nM T09960 C1PV5A 44590718 IC50 = 17.9 nM T09960 CU40QM 44590719 IC50 > 25000 nM T09960 C37QZC 44590720 IC50 = 0.003 nM T09960 CB32OD 44590738 IC50 = 313 nM T09960 CUQ63O 44590739 IC50 = 41 nM T09960 CDOP14 44590750 IC50 = 0.16 nM T09960 CRDP72 44590751 IC50 = 6430 nM T09960 CTLW28 44590752 IC50 = 3.16 nM T09960 CT92AQ 44590753 IC50 = 3.4 nM T09960 C3P7HB 44590798 IC50 = 3.63 nM T09960 CZ0C5N 44590799 IC50 = 4.83 nM T09960 CBAK64 44590800 IC50 = 25.3 nM T09960 C2L6AI 44590801 IC50 = 33.7 nM T09960 C9BPW4 44590849 IC50 = 102 nM T09960 CRQ09H 44590850 IC50 = 56 nM T09960 CPV4L8 44590862 IC50 = 64.4 nM T09960 CA79TX 44590863 IC50 = 73.5 nM T09960 CIH56J 44590864 IC50 = 2310 nM T09960 CZ5HT9 44590865 IC50 = 382 nM T09960 CAC12Y 44590943 IC50 = 540 nM T09960 C2EB4O 44590944 IC50 = 1849 nM T09960 CFE24S 44590945 IC50 = 21.4 nM T09960 CHQM54 44590946 IC50 = 94.6 nM T09960 C4N1MT 46191232 IC50 = 2 nM T09960 C1SAG3 46191233 IC50 < 0.3 nM T09960 CK3N1G 46206137 IC50 > 10000 nM T09960 CV2G0F 46225342 IC50 > 2500 nM T09960 C6V9JA 46225343 IC50 = 102 nM T09960 CSET80 46225344 IC50 = 59 nM T09960 CSX9I8 46225345 IC50 = 339 nM T09960 C5G3NW 46225346 IC50 = 167 nM T09960 C28WID 46225347 IC50 = 37 nM T09960 CZFT40 46225348 IC50 = 361 nM T09960 CIA1T4 46225349 IC50 = 46 nM T09960 CS4T3F 46225350 IC50 = 28 nM T09960 C2POI6 46225394 IC50 = 65 nM T09960 C6VCG0 46225395 IC50 = 55 nM T09960 CJ9R1Y 46225428 IC50 = 1943 nM T09960 C2E6PS 46225429 IC50 = 69 nM T09960 C1G8IP 46225512 IC50 = 27 nM T09960 CW8RZ6 46225513 IC50 = 56 nM T09960 CS1H4X 46225514 IC50 = 27 nM T09960 C3H6PF 46225515 IC50 = 10 nM T09960 CZL79B 46225526 IC50 = 30 nM T09960 CK56CR 46225527 IC50 = 38 nM T09960 CQJM47 46225528 IC50 = 5 nM T09960 CVX2D6 46225529 IC50 = 66 nM T09960 C6Q2ML 46225530 IC50 = 15 nM T09960 CC9J8S 46225531 IC50 = 53 nM T09960 CV2SG0 46225532 IC50 = 1 nM T09960 CIV7G4 46225533 IC50 = 3 nM T09960 CMA4Y5 46226118 IC50 = 10000 nM T09960 C1Z3BR 46226120 IC50 = 170 nM T09960 C09LCK 46226122 IC50 = 86 nM T09960 CX6PK2 46226124 IC50 = 79 nM T09960 CAF2T0 46226126 IC50 = 130 nM T09960 CB8Q4K 46226128 IC50 = 42 nM T09960 CP10VT 46226130 IC50 = 92 nM T09960 CF85BE 46226132 IC50 = 13 nM T09960 C3YQ7A 46837425 IC50 = 10000 nM T09960 C8K4CT 46837428 IC50 > 10000 nM T09960 C8VZ9P 46837429 IC50 > 10000 nM T09960 CAG58V 46837553 IC50 = 253 nM T09960 C2E4CD 46837554 IC50 = 10000 nM T09960 CPC64Z 46837555 IC50 > 10000 nM T09960 C7XG1V 46837556 IC50 > 10000 nM T09960 C0RF1D 46864993 IC50 = 18 nM T09960 COY59E 46866599 IC50 = 8 nM T09960 CHQI42 46880774 IC50 = 6 nM T09960 CEKG54 46880775 IC50 = 30 nM T09960 CTC2X7 46880847 IC50 = 38 nM T09960 CUG39Q 46880848 IC50 = 7 nM T09960 CH0M1Q 46880849 IC50 = 5 nM T09960 CEY3D2 46880850 IC50 = 13 nM T09960 C69OGT 46880887 IC50 = 5 nM T09960 C6TN7S 46882070 IC50 > 500 nM T09960 C1YG5B 46882071 IC50 > 500 nM T09960 C23WRH 46882072 IC50 > 500 nM T09960 CLA67N 46882073 IC50 = 92 nM T09960 C9AR5O 46882074 IC50 = 98 nM T09960 C1Z8YT 46882075 IC50 = 45 nM T09960 CYV6Z5 46882076 IC50 = 14 nM T09960 C8EV6W 46882077 IC50 = 15 nM T09960 C3SJ0I 46882078 IC50 = 25 nM T09960 C5AQ1Y 46882079 IC50 = 61 nM T09960 C6XOK3 46882080 IC50 = 44 nM T09960 CUNP07 46882081 IC50 = 34 nM T09960 CSH9R7 46882082 IC50 = 23 nM T09960 C2SZI3 46882083 IC50 = 27 nM T09960 C1K3TC 46882871 IC50 = 100 nM T09960 CC9VR6 46882872 IC50 = 18 nM T09960 CXEO65 46882873 IC50 = 24 nM T09960 C69SIF 46882916 IC50 = 10 nM T09960 CMP29J 46882947 IC50 = 7 nM T09960 C20IML 46882948 IC50 = 58 nM T09960 C2U9EO 46882985 IC50 = 100 nM T09960 C18KLW 46883025 IC50 = 61 nM T09960 C8I9ZQ 46883026 IC50 = 80 nM T09960 CO8Y6D 46883027 IC50 = 24 nM T09960 C7TO8G 46883028 IC50 = 22 nM T09960 CZ6CK2 46883029 IC50 = 12 nM T09960 CU32SF 46883030 IC50 = 97 nM T09960 CM9UG5 46883031 IC50 = 10 nM T09960 CG7OL0 46883507 IC50 = 51 nM T09960 CV14GK 46888453 IC50 = 6 nM T09960 CP45CJ 46888454 IC50 = 15 nM T09960 CC7KQ1 46888455 IC50 = 11 nM T09960 CK0X4C 46888456 IC50 = 7 nM T09960 C30THG 46888478 IC50 = 3 nM T09960 CAK75S 46888479 IC50 = 4 nM T09960 C63UBP 46888480 IC50 = 8 nM T09960 CG7HE8 46888496 IC50 = 18 nM T09960 CI8MG4 46888497 IC50 = 15 nM T09960 CPO0Z8 46888498 IC50 = 465 nM T09960 CQS95E 46888499 IC50 = 9 nM T09960 CP8YH4 46888524 IC50 = 14 nM T09960 CUY17G 46888525 IC50 = 6 nM T09960 CPI6N7 46888526 IC50 = 26 nM T09960 CGZX65 46888544 IC50 = 19 nM T09960 C3NXP5 46888545 IC50 = 7 nM T09960 CM0X6G 46888546 IC50 = 44 nM T09960 C79OQJ 46888563 IC50 = 14 nM T09960 C63YJU 46888564 IC50 = 30 nM T09960 CA45RF 46888565 IC50 = 12 nM T09960 CU2TE0 46888566 IC50 = 27 nM T09960 C2PJG4 46888581 IC50 = 20 nM T09960 C5ZQ2A 46888582 IC50 = 13 nM T09960 CBD19K 46888583 IC50 = 12 nM T09960 CDI40V 46888584 IC50 = 9 nM T09960 C0FL8H 46888604 IC50 = 25 nM T09960 CVD8K7 46888605 IC50 = 30 nM T09960 C7A2BS 46888606 IC50 = 34 nM T09960 CULC94 46890340 IC50 = 26 nM T09960 CRE91L 46890341 IC50 = 62 nM T09960 CV2RH7 46890342 IC50 = 20 nM T09960 C64DLQ 46890343 IC50 = 8 nM T09960 CI9MR8 46890345 IC50 > 500 nM T09960 CWY7D6 46890346 IC50 = 33 nM T09960 C5O8EZ 46890427 IC50 = 24 nM T09960 C2KJS7 46890428 IC50 = 12 nM T09960 CJ9SL0 46890429 IC50 = 25 nM T09960 C43QJG 49768639 IC50 = 31 nM T09960 CDM18G 49768863 IC50 = 1.4 nM T09960 C3E5JT 49798079 IC50 > 30 nM T09960 CZQ54K 49798080 IC50 = 6.15 nM T09960 C32OXR 49798081 IC50 = 220.6 nM T09960 CJ5GZ2 49798082 IC50 = 1.09 nM T09960 CUQ79L 49798083 IC50 = 20.2 nM T09960 C8RVJ9 49798084 IC50 = 37.7 nM T09960 C9W7HN 49798085 IC50 = 1.71 nM T09960 C1UKV9 49798086 IC50 = 2.66 nM T09960 CFGM47 49798087 IC50 = 3.2 nM T09960 CTA1U3 49798088 IC50 = 6.15 nM T09960 CQ3R2G 49798089 IC50 = 1.62 nM T09960 CAWQ56 49798090 IC50 = 1.69 nM T09960 C61NQS 49798129 IC50 = 3.5 nM T09960 C6VPR9 49798130 IC50 = 14.6 nM T09960 C20OMQ 49798131 IC50 = 5.3 nM T09960 C72VPW 49798132 IC50 = 11 nM T09960 C4EQ0K 49798133 IC50 = 3.6 nM T09960 CV8XW0 49798156 IC50 = 17.8 nM T09960 C4I0TN 49798157 IC50 = 149.2 nM T09960 CK5S2Z 49798158 IC50 = 4 nM T09960 CQVG17 49798349 IC50 = 630.96 nM T09960 CG83TP 49798920 IC50 = 320 nM T09960 C3Y1AN 49799705 IC50 = 81 nM T09960 C7M8DB 49799707 IC50 = 57 nM T09960 CIY75R 49799711 IC50 = 42 nM T09960 CH4JV5 49864967 IC50 = 318 nM T09960 C4RQ8B 49864968 IC50 = 30 nM T09960 C8ZFG4 49864969 IC50 = 8.85 nM T09960 CZ2LD9 49864970 IC50 = 38.3 nM T09960 C7GU4O 49864971 IC50 = 1.38 nM T09960 CV4UR2 49864972 IC50 = 11.17 nM T09960 C5HKC2 49864973 IC50 = 2.98 nM T09960 C74QMJ 49864974 IC50 = 6.77 nM T09960 C5I8KJ 49864975 IC50 = 11.4 nM T09960 CP4XR3 49864976 IC50 = 30 nM T09960 C7JF3Q 49864977 IC50 = 3.98 nM T09960 CZ7CR9 50915506 IC50 = 0.4 nM T09960 CI32TR 50992246 IC50 = 5.3 nM T09960 CF0A5Z 50992494 IC50 = 0.2 nM T09960 C4IFR9 50992499 IC50 < 0.1 nM T09960 CB1VU9 50992574 IC50 = 5 nM T09960 C3S5HO 50992575 IC50 = 3 nM T09960 C51FNM 50992577 IC50 = 0.4 nM T09960 C90LTR 50992639 IC50 = 0.4 nM T09960 CWOE69 50992640 IC50 = 0.4 nM T09960 CS5C4D 50992641 IC50 = 0.3 nM T09960 CFB75J 50992642 IC50 < 0.1 nM T09960 CFG8M7 50992643 IC50 < 0.1 nM T09960 C41QJN 50992719 IC50 < 0.1 nM T09960 C4BP6M 50992720 IC50 < 0.1 nM T09960 CIO9B5 50992721 IC50 < 0.1 nM T09960 C2ST3V 50992722 IC50 < 0.1 nM T09960 C0XF6H 50993435 IC50 = 29 nM T09960 CQJ83W 50993436 IC50 = 9 nM T09960 C51DPL 50993591 IC50 = 0.1 nM T09960 C2D4XS 50993592 IC50 = 0.6 nM T09960 C70BEM 50993593 IC50 = 0.2 nM T09960 C7RX0Y 52918140 IC50 = 20 nM T09960 C7BAV4 52940989 IC50 = 41 nM T09960 C5Z1PK 52941008 IC50 = 52 nM T09960 C36JTE 52941648 IC50 = 3.3 nM T09960 CI3C8V 52942058 IC50 = 137 nM T09960 CLO38X 52942071 IC50 = 19 nM T09960 C2G1RT 52942078 IC50 = 744 nM T09960 C8V2JI 52942223 IC50 = 420 nM T09960 C9G8VW 52943283 IC50 = 99 nM T09960 CZ10FK 52943389 IC50 = 4.5 nM T09960 C03XMU 52943390 IC50 = 4.5 nM T09960 C84OYJ 52943424 IC50 = 35 nM T09960 CX3LY2 52943425 IC50 = 3100 nM T09960 CAU0O1 52943426 IC50 = 150 nM T09960 C5BEV7 52944086 IC50 = 46 nM T09960 C86MFB 52944231 IC50 = 4123 nM T09960 CQ38KM 52944537 IC50 = 11 nM T09960 C9C5OP 52944586 IC50 = 15 nM T09960 C1ZPU9 52944587 IC50 = 6.9 nM T09960 CAC4V2 52944616 IC50 = 26 nM T09960 CM24UY 52944617 IC50 = 60 nM T09960 C91GLQ 52944618 IC50 = 210 nM T09960 C64CAT 52944644 IC50 = 313 nM T09960 C4KLV6 52945332 IC50 = 34 nM T09960 CIB1K6 52945865 IC50 = 87 nM T09960 CLAH27 52946506 IC50 = 8 nM T09960 CG8S9O 52946946 IC50 > 5000 nM T09960 CA7Z6L 52946953 IC50 > 5000 nM T09960 C1C5BV 52946954 IC50 = 1.2 nM T09960 C1X9RI 52947038 IC50 = 30 nM T09960 C0F1WE 52947044 IC50 = 63 nM T09960 C8CZL6 52947063 IC50 = 22 nM T09960 C6KCU2 52947064 IC50 = 64 nM T09960 CJZK15 52947090 IC50 = 34 nM T09960 CS9UX8 52947091 IC50 = 3.7 nM T09960 CKI5X6 52947100 IC50 > 5000 nM T09960 C1ZK2O 52947741 IC50 > 5000 nM T09960 CJT61Q 52947748 IC50 = 93 nM T09960 CZK6D2 52948162 IC50 = 2819 nM T09960 C64DXZ 52948248 IC50 > 5000 nM T09960 C0ZF7V 52948264 IC50 = 8.6 nM T09960 C6LV0Q 52948295 IC50 = 20.5 nM T09960 CX2QU9 52948296 IC50 = 2.6 nM T09960 CI5EM7 52949128 IC50 = 2173 nM T09960 COH5M1 52949523 IC50 = 27 nM T09960 CU0P3Q 52949553 IC50 = 65 nM T09960 CU25FT 52949601 IC50 = 2832 nM T09960 C70QNI 53260398 IC50 = 0.3548 nM T09960 C7U1ZC 53317132 IC50 > 1000 nM T09960 C0AS8E 53318853 IC50 = 77 nM T09960 C8K5QI 53318854 IC50 = 572 nM T09960 CLP07M 53319405 IC50 = 2 nM T09960 CCV39H 53319838 IC50 = 4.6 nM T09960 CH34SY 53319839 IC50 > 1000 nM T09960 C76HPL 53321427 IC50 = 22.5 nM T09960 C1HOS5 53321482 IC50 = 312 nM T09960 CK2M9J 53321616 IC50 = 18 nM T09960 CK2JD6 53322809 IC50 = 108 nM T09960 C35XLW 53322810 IC50 = 34.8 nM T09960 C4EV2O 53323818 IC50 > 1000 nM T09960 CH3LK8 53324139 IC50 > 1000 nM T09960 COYC36 53324140 IC50 = 546 nM T09960 C48XCJ 53324141 IC50 = 206 nM T09960 CO93PA 53324304 IC50 = 23 nM T09960 CC1ER2 53324598 IC50 = 181.97 nM T09960 C9B7FY 53325088 IC50 = 211 nM T09960 C9YGA3 53325385 IC50 = 370 nM T09960 CM12CJ 53325460 IC50 = 11.1 nM T09960 CY15EU 53325639 IC50 = 26.5 nM T09960 CYA3F1 53325983 IC50 = 0.5 nM T09960 CD1SK7 53326700 IC50 = 1000 nM T09960 C8E0DF 53326701 IC50 = 204 nM T09960 C7PQ1Y 53326702 IC50 = 201 nM T09960 C8C7PV 53389082 IC50 = 4600 nM T09960 C9QD2Z 53389084 IC50 = 10010 nM T09960 CC8ME1 53389637 IC50 = 275.42 nM T09960 C13SIB 53389710 IC50 = 512.86 nM T09960 CXW05M 53389845 IC50 = 575.44 nM T09960 CS0Q8N 53389902 IC50 = 213.8 nM T09960 C4OL5J 54580080 IC50 = 2238.72 nM T09960 CL4N5M 54580081 IC50 = 19.95 nM T09960 C0O5LX 54580082 IC50 = 251.19 nM T09960 CFEK69 54580093 IC50 = 177.83 nM T09960 CRV8T5 54580467 IC50 = 40 nM T09960 C8RK1D 54580468 IC50 = 120 nM T09960 CTO38W 54580469 IC50 = 220 nM T09960 CIW93N 54581068 IC50 = 2511.89 nM T09960 CI93ZC 54581069 IC50 > 3162.28 nM T09960 CS3PM2 54581070 IC50 = 1584.89 nM T09960 C80DUA 54581071 IC50 = 1995.26 nM T09960 C05GIL 54581076 IC50 = 17.78 nM T09960 C8VQU5 54581478 IC50 = 12250 nM T09960 CU8N4Z 54581479 IC50 = 30 nM T09960 C9X4EW 54581480 IC50 = 140 nM T09960 C2AVP1 54582104 IC50 = 257.04 nM T09960 C8SEU2 54582105 IC50 = 10 nM T09960 CX0WM5 54582110 IC50 = 15.85 nM T09960 CUWR02 54583048 IC50 > 3162.28 nM T09960 CCO15Z 54583049 IC50 = 1778.28 nM T09960 CML64U 54583458 IC50 = 290 nM T09960 C6H4BZ 54583459 IC50 = 21370 nM T09960 CCRX35 54583460 IC50 = 30 nM T09960 C49QZJ 54583462 IC50 = 3800 nM T09960 CEAG79 54584051 IC50 > 3162.28 nM T09960 C53YSX 54584052 IC50 = 398.11 nM T09960 CS2UN4 54584053 IC50 = 100 nM T09960 C96PFQ 54584058 IC50 = 31.62 nM T09960 C7CAN9 54584059 IC50 = 5.012 nM T09960 C5NRH1 54584427 IC50 = 970 nM T09960 CTRG70 54585004 IC50 > 3162.28 nM T09960 CHPB98 54585369 IC50 = 1760 nM T09960 CP8Q6M 54585383 IC50 = 5620 nM T09960 CH7NT9 54585384 IC50 = 130 nM T09960 CI1U4V 54585385 IC50 = 3390 nM T09960 C9ONK2 54585963 IC50 = 251.19 nM T09960 CQP1B8 54585964 IC50 = 8.913 nM T09960 CB82XJ 54585972 IC50 > 3162.28 nM T09960 CGS76T 54586286 IC50 = 180 nM T09960 CW97CT 54586339 IC50 = 100 nM T09960 CEA41I 54587374 IC50 = 17010 nM T09960 C7PHF2 54752872 IC50 = 10100 nM T09960 CVA1S8 54752874 IC50 = 9200 nM T09960 CG4U7M 54753646 IC50 = 5400 nM T09960 CM0Z8W 56647023 IC50 = 6.9 nM T09960 CYR89T 56647076 IC50 = 6.4 nM T09960 C57DEP 56657984 IC50 = 59000 nM T09960 CWF8C3 56657986 IC50 = 180000 nM T09960 C1K5GS 56659271 IC50 = 48090 nM T09960 CGK57R 56661522 IC50 = 81000 nM T09960 CMV8C3 56661524 IC50 = 25000 nM T09960 CZN3H8 56661526 IC50 = 20000 nM T09960 C2BMX7 56661530 IC50 = 1148000 nM T09960 C48GTM 56664935 IC50 = 50000 nM T09960 CKQG84 56664937 IC50 = 23000 nM T09960 CA9ML1 56664939 IC50 = 190000 nM T09960 CFYI08 56668364 IC50 = 270000 nM T09960 C4TXR2 56669615 IC50 = 7800 nM T09960 CJC18T 56671869 IC50 = 120000 nM T09960 CNX6F5 56673133 IC50 = 15240 nM T09960 CXI8E3 56675256 IC50 = 140000 nM T09960 C5U1RV 56676454 IC50 = 37610 nM T09960 CGS0W3 56678574 IC50 = 23000 nM T09960 CGS5P2 56678576 IC50 = 21000 nM T09960 CUL60G 56678578 IC50 = 35000 nM T09960 C5LJ8C 56681915 IC50 = 5200 nM T09960 COS02D 56681917 IC50 = 3900 nM T09960 C3A7OC 56683102 IC50 = 8400 nM T09960 CHM6Z8 56750906 IC50 = 36000 nM T09960 CQ9S6H 56754672 IC50 = 70000 nM T09960 C97HKS 57331246 IC50 > 1000 nM T09960 CR3HF8 57331274 IC50 = 25.73 nM T09960 CXV90D 57331275 IC50 = 76.03 nM T09960 CFC2Q4 57331276 IC50 = 35.47 nM T09960 C50UMI 57331277 IC50 = 320.33 nM T09960 C9Y6MI 57331278 IC50 = 25.53 nM T09960 CVDQ59 57331304 IC50 = 64.07 nM T09960 C6VUQ9 57331305 IC50 = 525 nM T09960 C36BJH 57331306 IC50 = 93.53 nM T09960 CV7X0G 57331307 IC50 = 26.37 nM T09960 CX58OH 57331308 IC50 = 473.33 nM T09960 C5JFZ1 57331339 IC50 = 75.3 nM T09960 CXO80S 57331340 IC50 = 202.43 nM T09960 CNS7H5 57335017 IC50 = 7300 nM T09960 CBF53W 57384005 IC50 = 0.3 nM T09960 CF1OM2 57384006 IC50 = 0.3 nM T09960 C16ZHL 57390535 IC50 = 8 nM T09960 CZOY39 57391591 IC50 = 810 nM T09960 CCA7D3 57391720 IC50 = 8.9 nM T09960 C5ND1L 57391721 IC50 = 0.44 nM T09960 C5QD2I 57391722 IC50 = 0.55 nM T09960 CCKJ07 57392302 IC50 = 387 nM T09960 C0YX7L 57392303 IC50 = 0.7 nM T09960 CK59VA 57392726 IC50 = 2850 nM T09960 CPQC75 57393451 IC50 = 3.5 nM T09960 CO29JI 57394057 IC50 = 1.6 nM T09960 C3F4XE 57394058 IC50 = 7 nM T09960 CGV90O 57395178 IC50 = 3.1 nM T09960 C9G6OJ 57395179 IC50 = 5 nM T09960 CGR9F3 57395184 IC50 < 0.1 nM T09960 CSH0P9 57395816 IC50 = 12.3 nM T09960 C3AB8V 57395817 IC50 = 1.5 nM T09960 C23QVB 57395818 IC50 = 130 nM T09960 CVXD20 57396843 IC50 = 5.4 nM T09960 C75SYT 57396949 IC50 = 229 nM T09960 CWU1I0 57396950 IC50 < 0.1 nM T09960 CR41GU 57396951 IC50 = 3700 nM T09960 C9YT0S 57396952 IC50 = 0.69 nM T09960 CTH3P5 57396953 IC50 < 0.1 nM T09960 C0R1ET 57397595 IC50 = 116 nM T09960 C23IKA 57397596 IC50 = 11 nM T09960 CZ29HN 57397597 IC50 = 3 nM T09960 CC72RQ 57397598 IC50 = 2.4 nM T09960 CH58PW 57397603 IC50 = 1586 nM T09960 CA2IY7 57398009 IC50 = 1300 nM T09960 CK97BJ 57400372 IC50 = 39 nM T09960 C19SNT 57400373 IC50 = 162 nM T09960 CA5KO3 57400374 IC50 = 1.1 nM T09960 CT31JR 57400375 IC50 = 794 nM T09960 C0H7ME 57401041 IC50 = 90 nM T09960 CCJ1I2 57401042 IC50 = 12 nM T09960 C5NDS6 57402175 IC50 = 1.6 nM T09960 CRUX38 57402798 IC50 = 50 nM T09960 CV96NF 57402799 IC50 = 3 nM T09960 C9ER8K 57402800 IC50 = 2 nM T09960 C37NBY 57402801 IC50 = 0.09 nM T09960 CA7TX2 57402802 IC50 = 0.98 nM T09960 CXYB90 57403173 IC50 = 1000 nM T09960 CU4S6M 57403931 IC50 = 15 nM T09960 CC0D8X 57403932 IC50 = 0.68 nM T09960 CHJ87A 57656833 IC50 = 22 nM T09960 CZ71SN 58282592 IC50 = 650 nM T09960 C0YWT1 58509213 IC50 > 10000 nM T09960 C6JKM0 58834906 IC50 = 0.6 nM T09960 CR8L7P 58834946 IC50 = 0.9 nM T09960 CF9Z0L 58834953 IC50 = 1.1 nM T09960 CMJ59Z 58834969 IC50 = 0.4 nM T09960 CM6Z7S 58835000 IC50 = 1.3 nM T09960 C4PWA9 58835024 IC50 = 1.4 nM T09960 C7RXU8 58835027 IC50 = 1.3 nM T09960 CC36OU 58835113 IC50 = 0.9 nM T09960 C2XRL5 58835114 IC50 = 1.1 nM T09960 CN3RD2 58835155 IC50 = 1.5 nM T09960 CCR4T7 58835217 IC50 = 0.7 nM T09960 C76HQB 59458061 IC50 = 0.4 nM T09960 C5KUQ8 59458103 IC50 = 1.7 nM T09960 CEI9H7 59458159 IC50 = 8.6 nM T09960 CQTK25 59458213 IC50 = 5.3 nM T09960 C46UHJ 59458228 IC50 = 0.4 nM T09960 C7SOK2 59458245 IC50 = 1 nM T09960 C27NIL 59458247 IC50 = 0.9 nM T09960 C6GPD8 59959034 IC50 = 1 nM T09960 CT0NG6 62706106 IC50 = 0.7 nM T09960 CKA9V2 62706107 IC50 = 0.11 nM T09960 CB91CU 62706108 IC50 = 0.9 nM T09960 CG58WC 62706109 IC50 = 0.8 nM T09960 CA4RU3 62706110 IC50 = 0.3 nM T09960 C0N8XJ 62707281 IC50 = 9200 nM T09960 CHU5Q0 62707283 IC50 = 16300 nM T09960 CJ2S6W 62707285 IC50 > 100000 nM T09960 CTC5D7 62707286 IC50 > 30000 nM T09960 C9NGJ8 62707287 IC50 = 6500 nM T09960 C40ORM 62707443 IC50 = 7800 nM T09960 CX4MO7 62707444 IC50 = 10000 nM T09960 CF4X6H 62707445 IC50 = 8400 nM T09960 CPDZ56 62707446 IC50 = 4600 nM T09960 C2N9YG 62707447 IC50 = 48100 nM T09960 C3X8YK 62707448 IC50 = 15200 nM T09960 CAY3H7 62707598 IC50 = 37600 nM T09960 CQR25M 66767933 IC50 = 321 nM T09960 CO62SG 66768099 IC50 = 137 nM T09960 CC81NU 66768640 IC50 = 1242 nM T09960 CCB1T5 68764898 IC50 = 2.4 nM T09960 C5O0JN 68764925 IC50 = 3 nM T09960 C70QJS 68767049 IC50 = 3.4 nM T09960 C8VU1C 68767078 IC50 = 22 nM T09960 C2YRL3 68769802 IC50 = 18 nM T09960 C39SPK 68772423 IC50 = 190 nM T09960 CV8E4C 69696607 IC50 = 750000 nM T09960 CDF0Q5 69697526 IC50 = 640000 nM T09960 C0POJ4 70685193 IC50 = 400 nM T09960 CU62NM 70688699 IC50 = 16400 nM T09960 CQOD53 70690765 IC50 = 10500 nM T09960 CZ0Y7T 70692897 IC50 > 30000 nM T09960 C1ACG8 70692902 IC50 = 9200 nM T09960 CW6UA5 70694934 IC50 > 30000 nM T09960 CV10AS 70694935 IC50 > 30000 nM T09960 CV53PW 70694941 IC50 = 13700 nM T09960 CW0B9M 71451541 IC50 = 31.1 nM T09960 C0F7NL 71451877 IC50 = 0.17 nM T09960 CDJN04 71458736 IC50 = 1.2 nM T09960 CP2UK0 71458737 IC50 = 14.3 nM T09960 CIP7D8 71462570 Ki = 1 nM T09960 CI8Q1K 71717723 Ki = 31 nM T09960 CP5NQ2 71718331 Ki = 210 nM T09960 CZ5C6V 71718930 Ki = 150 nM T09960 CC8JQ9 71719547 Ki = 50 nM T09960 C8CB3S 72711047 IC50 = 2.5 nM T09960 CIV83U 72711048 IC50 = 15 nM T09960 CFY8W4 72711049 IC50 = 34.8 nM T09960 CZG4V5 72711050 IC50 = 157.6 nM T09960 C8E2FK 72711051 IC50 = 700.8 nM T09960 CA5B9Z 72711277 IC50 = 4.7 nM T09960 C4UJW6 72711278 IC50 = 7.1 nM T09960 CGT0X3 72711279 IC50 = 832 nM T09960 CZI06T 72711280 IC50 = 300.7 nM T09960 C7XS9L 72711281 IC50 = 117.1 nM T09960 CM0OT6 72711506 IC50 = 24.7 nM T09960 C4HG7X 72711507 IC50 = 6.4 nM T09960 CTG02P 72711508 IC50 = 3.6 nM T09960 C37CFT 72711739 IC50 = 0.9 nM T09960 C7Q6PX 72711740 IC50 = 0.8 nM T09960 C8BG4M 72711741 IC50 = 0.9 nM T09960 C86FZB 72711742 IC50 = 1.2 nM T09960 CI0ZP4 72711955 IC50 = 5.9 nM T09960 CKR7P1 72711956 IC50 = 1.2 nM T09960 CHR42S 72711958 IC50 = 0.8 nM T09960 CMUB57 72712158 IC50 = 56 nM T09960 C6ISW8 72712159 IC50 = 12.4 nM T09960 C95SNW 72712160 IC50 = 169 nM T09960 CFAM28 72712161 IC50 = 17.9 nM T09960 C4MN3V 72712371 IC50 = 43.5 nM T09960 C6HR8T 72712372 IC50 = 279.5 nM T09960 C4Q2FZ 72712373 IC50 = 15.2 nM T09960 CT30UZ 72712374 IC50 = 50.7 nM T09960 C4ZSH1 72712375 IC50 > 1000 nM T09960 C9BK3P 72712597 IC50 = 15.8 nM T09960 C4ZFJ9 72712598 IC50 = 0.3 nM T09960 C0L2NB 72713858 IC50 = 39 nM T09960 C5VP8L 72713859 IC50 = 65.7 nM T09960 C1PO6A 72713860 IC50 = 13.6 nM T09960 CQ27VU 72713861 IC50 = 9039 nM T09960 CUI40C 72714076 IC50 = 14 nM T09960 C4ZRE2 72714077 IC50 = 1465 nM T09960 C4G1OR 72714078 IC50 = 1.2 nM T09960 C3Z7NO 72714079 IC50 = 1.5 nM T09960 CLA8B7 72714317 IC50 = 1702 nM T09960 C5MOY1 72714318 IC50 = 91 nM T09960 C9KB5E 72714319 IC50 = 195 nM T09960 CWY19V 72714320 IC50 = 11.7 nM T09960 C9XOJ0 72714321 IC50 = 10.4 nM T09960 CSV58N 73345281 Ki = 30000 nM T09960 CXD8A1 73346388 IC50 = 9.6 nM T09960 C82YDH 73346389 IC50 = 7.5 nM T09960 CNPK53 73346454 IC50 = 70800 nM T09960 CM19JQ 73346460 IC50 = 115000 nM T09960 C5XW1B 73346461 IC50 = 61000 nM T09960 CUQ94P 73346462 IC50 = 47000 nM T09960 CCJ01L 73347894 IC50 = 3.4 nM T09960 C6LTC1 73347956 IC50 = 77000 nM T09960 CMK7G0 73347961 IC50 = 63000 nM T09960 CR54VT 73349498 IC50 = 45000 nM T09960 C2TN1Z 73349499 IC50 = 65700 nM T09960 CA3X1K 73349500 IC50 = 88100 nM T09960 C4UP2I 73349506 IC50 = 56000 nM T09960 CO7ZS8 73349882 Ki = 5100 nM T09960 C1RV2N 73351054 IC50 = 138000 nM T09960 CFH03E 73351055 IC50 = 90000 nM T09960 CZ4C1R 73351059 IC50 = 28000 nM T09960 CFC9T7 73351060 IC50 = 51800 nM T09960 CD20KR 73352463 IC50 = 12.7 nM T09960 COGK67 73352528 IC50 = 92200 nM T09960 C04HGN 73352529 IC50 = 61000 nM T09960 C4D1TK 73352534 IC50 = 59000 nM T09960 CZWL45 73353307 EC50 = 0.18 nM T09960 C1MK9E 73354018 IC50 = 66200 nM T09960 C9TQ1F 73355478 IC50 = 22.5 nM T09960 CHKD46 73355549 IC50 = 77800 nM T09960 C2G5NZ 73355550 IC50 = 28700 nM T09960 C98NGO 73355552 IC50 = 73000 nM T09960 C0O3UA 73355553 IC50 = 38800 nM T09960 C9URF8 73355554 IC50 = 43500 nM T09960 C84QWC 73357100 IC50 = 64000 nM T09960 C8PJU5 76308345 IC50 = 599.79 nM T09960 CJPW31 76308985 IC50 = 1499.68 nM T09960 C82LXO 76308986 IC50 = 34.99 nM T09960 CV73GF 76309037 IC50 = 100 nM T09960 CHEU38 76310164 IC50 = 86.7 nM T09960 C3W7VP 76310165 IC50 = 151.8 nM T09960 C6JAT5 76311990 IC50 = 399.94 nM T09960 C58AGV 76312665 IC50 = 209.89 nM T09960 C5J6YC 76312666 IC50 = 57.02 nM T09960 C7WO1R 76313867 IC50 = 251.67 nM T09960 COZM91 76315543 IC50 = 1000 nM T09960 CF20LV 76315544 IC50 = 6998.42 nM T09960 C1EV0K 76316185 IC50 = 10.99 nM T09960 CS3BE1 76316241 IC50 = 1.995 nM T09960 CA72FV 76316242 IC50 = 39.81 nM T09960 CZ6L7V 76316949 IC50 = 14.4 nM T09960 C3QU8F 76317388 IC50 = 125.81 nM T09960 C20DSV 76317476 IC50 = 27 nM T09960 C24QYM 76317477 IC50 > 1000 nM T09960 C5TW0Z 76319890 IC50 = 169.82 nM T09960 CRN39I 76319891 IC50 = 3698.28 nM T09960 CHJ74V 76319944 IC50 = 1000 nM T09960 C9TEP7 76321110 IC50 > 1000 nM T09960 C9IZV4 76321206 IC50 = 3 nM T09960 C7QA1M 76322864 IC50 = 1000 nM T09960 CI97JM 76323541 IC50 = 1399.59 nM T09960 CTW39E 76324825 IC50 = 2.6 nM T09960 CL92XF 76324826 IC50 = 360 nM T09960 CH60RK 76327118 IC50 = 839.46 nM T09960 CL5Y7P 76327119 IC50 = 599.79 nM T09960 CFY46V 76327120 IC50 = 100 nM T09960 CG81BM 76327166 IC50 = 0.7943 nM T09960 CPR37U 76327885 IC50 = 112 nM T09960 CPV7L2 76330768 IC50 = 449.78 nM T09960 CLJ7E0 76330769 IC50 = 319.89 nM T09960 CFR3L2 76330770 IC50 = 46.99 nM T09960 CFLJ46 76330829 IC50 = 0.7586 nM T09960 CKA2Z8 76334365 IC50 = 1000 nM T09960 C8DW4B 76335572 IC50 = 196.9 nM T09960 C8ENW7 76335673 IC50 = 0.96 nM T09960 C03MUJ 86294766 IC50 = 48000 nM T09960 CI67KS 89702731 IC50 = 126 nM T09960 CH58FP 90656325 IC50 = 10300 nM T09960 C89GMZ 90656326 IC50 = 6450 nM T09960 CRFE08 90656327 IC50 > 50000 nM T09960 CV1DY8 90656328 IC50 = 16800 nM T09960 C5UW7K 90656329 IC50 > 50000 nM T09960 CZN8T2 90656330 IC50 = 6290 nM T09960 C7B2PH 90656331 IC50 > 50000 nM T09960 CPY6G0 90656332 IC50 > 50000 nM T09960 CPZ46K 90656333 IC50 = 23000 nM T09960 CAYE46 90656334 IC50 = 9800 nM T09960 C0KCP6 90656335 IC50 = 41200 nM T09960 C37ZBS 90656336 IC50 > 50000 nM T09960 CP5X4Y 90656337 IC50 = 45800 nM T09960 CEH42L 90656338 IC50 = 45900 nM T09960 CYX8F5 90656339 IC50 = 27000 nM T09960 C21GTQ 90656340 IC50 = 19800 nM T09960 C2NWY9 90656341 IC50 = 5100 nM T09960 CQ95YH 90656342 IC50 = 25600 nM T09960 C0LYS7 90656343 IC50 = 28100 nM T09960 C24AMG 90664936 IC50 = 35 nM T09960 CY8E3J 90665058 IC50 = 21 nM T09960 CYP01O 90665176 IC50 = 71 nM T09960 CJ2ME7 90666577 IC50 = 622 nM T09960 CEA06F 90666578 IC50 = 14.2 nM T09960 CIY0P6 90666579 IC50 = 1570 nM T09960 CI53XQ 90666580 IC50 = 7910 nM T09960 C3L6KU 91820689 IC50 = 3 nM T09960 C6ENV5 100951623 EC50 > 10000 nM T09960 CFRK67 118727171 IC50 = 8.3 nM T09960 C0LC6G 118727172 IC50 = 15.1 nM T09960 CIY59U 118727173 IC50 = 25.1 nM T09960 CL4H7J 118727174 IC50 = 6.6 nM T09960 C53EMI 118727175 IC50 = 30.1 nM T09960 C6J4DP 118727176 IC50 = 11.7 nM T09960 CYR91T 118727177 IC50 = 319.9 nM T09960 CZ20TS 118727178 IC50 = 25.1 nM T09960 C68DNS 118727179 IC50 = 30 nM T09960 CM67QT 118727180 IC50 = 10.9 nM T09960 CV1R5P 118727181 IC50 = 2158 nM T09960 C45PVA 118727182 IC50 = 204.1 nM T09960 C5KJW2 118727183 IC50 = 259.7 nM T09960 C03FHC 118727184 IC50 = 17.1 nM T09960 CGW9I8 118727185 IC50 = 33.2 nM T09960 CP57BR 118727186 IC50 = 8.8 nM T09960 CV5MD3 118727187 IC50 = 906 nM T09960 CJO04D 118727188 IC50 = 49.9 nM T09960 C8F6AV 118727189 IC50 = 3 nM T09960 C16VCE 118727190 IC50 = 239.5 nM T09960 C4E7QF 118727191 IC50 = 163.8 nM T09960 CXM94Y 118727192 IC50 = 6290 nM T09960 C5L3SI 122185608 IC50 = 12700 nM T09960 CQ5WN1 122185610 IC50 = 17300 nM T09960 CSR65M 122185612 IC50 = 12900 nM T09960 CWG5Y3 122185614 IC50 = 30100 nM T09960 CWV1B6 122185616 IC50 = 26800 nM T09960 C9FND3 122185618 IC50 = 38500 nM T09960 CV8H0G 122185620 IC50 = 46200 nM T09960 C57TSL 122185622 IC50 = 121500 nM T09960 C1XDO2 122185624 IC50 = 67700 nM T09960 C6X1JP 122185626 IC50 = 80900 nM T09960 CR3MI5 122185628 IC50 = 101200 nM T09960 CEL59A 122185630 IC50 = 173900 nM T09960 C0Z4RT 122185632 IC50 = 19300 nM T09960 C5L7KA 122185634 IC50 = 69000 nM T09960 CK67LU 122185636 IC50 = 23900 nM T09960 C2G7TC 122185638 IC50 = 18700 nM T09960 CD1MG8 122185640 IC50 = 1350 nM T09960 C60LPW 122668161 IC50 = 51.7 nM T09960 C4KQS3 122668167 IC50 = 33 nM T09960 C85JKN 122668190 IC50 = 3.1 nM T09960 C5DUQ7 122668213 IC50 = 2.6 nM T09960 C8T9ON 126567253 IC50 = 15.8 nM T09960 CTAG09 126567264 IC50 = 2.8 nM T09960 CFWG31 126567273 IC50 = 82.6 nM T09960 CN68LA 126567277 IC50 = 12 nM T09960 CK36LH 126567281 IC50 = 27.1 nM T09960 CUFI59 126567286 IC50 = 6.8 nM T09960 C5QT4N 126567306 IC50 = 9.1 nM T09960 CK73PJ 129907953 EC50 = 42460 nM T09960 CS4M1X 129908109 EC50 = 29670 nM T09960 C8QYG0 129908110 EC50 = 11220 nM T09960 CGD5O4 129908111 EC50 = 18850 nM T09960 C0PH6K 129908112 EC50 > 50000 nM T09960 C7WXL1 129908179 EC50 > 50000 nM T09960 C8P9OC 129908195 EC50 = 15990 nM T09960 CNC2W3 129908196 EC50 = 22840 nM T09960 C14IAU 129908213 EC50 > 50000 nM T09960 CE80MX 129908214 EC50 > 50000 nM T09960 C6N0SF 129908215 EC50 > 50000 nM T09960 CG1M2A 129908240 EC50 > 50000 nM T09960 CJS4A1 129908281 EC50 = 4850 nM T09960 C2QSU0 129908301 EC50 = 16250 nM T09960 C2U4JE 129908428 EC50 = 16560 nM T09960 CV72QT 129908452 EC50 = 16830 nM T09960 CAX21P 129908453 EC50 = 18770 nM T09960 CSG86U 129908454 EC50 = 23140 nM T09960 C17ZKU 129908455 EC50 = 30630 nM T09960 CY9MZ7 129908456 EC50 = 18340 nM T09960 CONW96 129908557 EC50 > 50000 nM T09960 C2YB7V 129908558 EC50 = 36300 nM T09960 CC9S4Q 129908559 EC50 > 200000 nM T09960 C5WGK9 129908560 EC50 = 55370 nM T09960 CSD1X5 132572938 EC50 > 10 nM T09960 CV8N7E 137635442 EC50 > 10 nM T09960 C52MBZ 137638300 EC50 > 10 nM T09960 CL8P3K 137641868 EC50 > 10 nM T09960 CR2HZ3 137648323 EC50 > 10 nM T09960 C2WT5B 137654404 EC50 > 10 nM T09960 C0X5EI 137655931 EC50 > 10 nM T09960 CYV7M3 137660245 EC50 = 2470 nM T09960 C32SJE 145961982 IC50 = 660 nM T09960 C56KSZ 145967247 IC50 = 1.288 nM T09960 CXA2G0 145967391 IC50 = 1100 nM T09960 C1SQ3H 145982775 IC50 = 2.9 nM T09960 CY0S1F 145983098 IC50 = 296.4 nM T09960 CCHZ83 145983159 IC50 = 24.5 nM T09960 C87XGI 145983513 IC50 = 16.2 nM T09960 CTRV17 145983733 IC50 = 2.9 nM T09960 CVD12G 145983844 IC50 = 20.6 nM T09960 CS26EW 145984103 IC50 = 87.9 nM T09960 CQ5EN9 145984502 IC50 = 2.6 nM T09960 C2ANL3 145984591 IC50 = 4 nM T09960 C50AOD 145984717 IC50 = 5.4 nM T09960 C4HAP0 145984727 IC50 = 2.3 nM T09960 C53PGI 145984829 IC50 = 2.6 nM T09960 C5IZJ6 145985042 IC50 = 2.9 nM T09960 C6YW8A 145985237 IC50 = 8.1 nM T09960 CYG9S8 145985461 IC50 = 2.8 nM T09960 CQOR04 145985672 IC50 = 3 nM T09960 C0JOG7 145985889 IC50 = 5.2 nM T09960 C4LA2T 145985894 IC50 = 9.7 nM T09960 CB0FC5 145986021 IC50 = 2.3 nM T09960 CP2Z5X 145986145 IC50 = 4.7 nM T09960 CNC59J 145986205 IC50 = 251.6 nM T09960 CAF10K 145986277 IC50 = 6.8 nM T09960 CFN4J8 145996522 EC50 = 4.467 nM T09960 CXT09R 154572822 IC50 = 287 nM T09960 COP6C1 155491018 EC50 = 5 nM T09960 CVQ31N 155513284 IC50 = 371.54 nM T09960 C86OHR 155529593 IC50 = 3469 nM T09960 CVS37C 155531379 IC50 = 1570 nM T09960 CZ04TG 155540798 IC50 = 323.59 nM T09960 C80LBZ 155554273 IC50 = 123.03 nM T09960 D01LRC 6479877 IC50 = 5400 nM T09960 D06MBD 11176403 IC50 < 3000 nM T09960 D06QRP 5311123 Ki = 66 nM T09960 D06XIC 6480205 IC50 = 9000 nM T09960 D06XRS 4716524 IC50 = 1099.01 nM T09960 D0BD3G 11188669 IC50 = 1000 nM T09960 D0BD6A 10278617 IC50 = 5.1 nM T09960 D0E4YP 9873888 Ki = 1.4 nM T09960 D0I3IZ 11267381 IC50 = 1700 nM T09960 D0J3BT 16663418 IC50 = 3.5 nM T00477 D0M8AB 750 Ki = 366000 nM T00477 D0X9RY 243 IC50 > 10000000 nM T00477 CFR5J9 6918 IC50 = 8213000 nM T00477 CL70CJ 13650 IC50 > 10000000 nM T00477 CVGZ72 14463 Ki = 11000 nM T00477 CJ49VP 352208 IC50 > 10000000 nM T00477 C49KEP 447315 IC50 = 2820000 nM T00477 CK97ZC 637090 IC50 > 10000000 nM T00477 CP58OT 637541 IC50 = 8386000 nM T00477 C79CFS 770980 IC50 = 5282000 nM T00477 CC6G4J 833670 IC50 > 5000000 nM T00477 CC31OH 1105076 Ki = 1500000 nM T00477 C9VNH4 2063443 IC50 = 5015000 nM T00477 C0GJ3Y 2113906 IC50 > 10000000 nM T00477 CO1V8G 2512481 IC50 = 5723000 nM T00477 CK7LH9 2905941 Ki = 1700000 nM T00477 C51QOE 3686650 IC50 = 5159000 nM T00477 CU68IK 7141881 IC50 > 100000 nM T00477 C90XSD 7535844 IC50 = 140000 nM T00477 COR2F1 11575956 Ki = 320000 nM T00477 C50VWH 11834812 Ki > 10000000 nM T00477 C5EJS6 11964443 Ki = 610000 nM T00477 CT68FK 89717779 IC50 = 630000 nM T00477 CKW4U0 89717825 IC50 = 520000 nM T00477 CFOH54 122190495 Ki = 1500000 nM T00477 C7P4VG 122190496 Ki = 4500000 nM T00477 C6IQO2 145978550 IC50 = 836000 nM T00477 D08JNG 867 Ki = 33000 nM T00477 D08ZAO 14925 Ki = 1300000 nM T02562 D03RTS 2662 IC50 = 425 nM T02562 D05DVP 5717 IC50 = 18100 nM T02562 D09JUG 60490 IC50 = 600 nM T02562 D0R1RS 3715 IC50 = 40600 nM T02562 D0Z5IU 1548887 IC50 = 80000 nM T02562 D07SDQ 969516 IC50 = 300 nM T02562 D0U2BH 65064 IC50 = 1800 nM T02562 D0F8KE 71059525 IC50 = 0.94 nM T02562 D0LY6S 71766655 IC50 = 3.56 nM T02562 D05HSW 3218 IC50 = 200 nM T02562 D09BKE 4553 IC50 = 10000 nM T02562 D0K2ER 3651377 IC50 = 3 nM T02562 D0N1SU 133021 EC50 = 100 nM T02562 CPW9G5 65126 IC50 = 5000 nM T02562 C2FLZ8 65751 IC50 = 430 nM T02562 C2H0JD 68066 IC50 = 1150 nM T02562 C0D2ZM 105049 IC50 = 2400 nM T02562 CF2O4N 158143 IC50 = 3000 nM T02562 C83FUH 159969 IC50 = 1100 nM T02562 CW8K1N 168928 IC50 = 5000 nM T02562 CQY9S5 174857 IC50 = 430 nM T02562 CS4HK9 295563 IC50 = 3700 nM T02562 CM6G9N 334102 IC50 = 9500 nM T02562 C0GPV1 402434 IC50 = 1300 nM T02562 C5CSG4 402435 IC50 = 1100 nM T02562 CNBQ26 402705 IC50 = 917 nM T02562 CUW26R 423227 IC50 = 400 nM T02562 C8P3CK 427265 IC50 = 500 nM T02562 C9K5UB 441677 IC50 = 1100 nM T02562 CLV4X1 442009 IC50 = 5000 nM T02562 CVO51F 591238 IC50 = 1150 nM T02562 C27XBF 610243 IC50 = 6700 nM T02562 CJ2WX9 622124 IC50 = 10400 nM T02562 CPL20I 973124 IC50 = 58 nM T02562 C8ULB6 994643 IC50 = 13600 nM T02562 CM20VO 995223 IC50 = 5400 nM T02562 CE4HM8 1032885 IC50 = 3000 nM T02562 C5GPB3 1076642 IC50 = 5100 nM T02562 CK6DV3 1082140 IC50 = 33 nM T02562 CF8GU3 1100244 IC50 = 4.6 nM T02562 C5ZF8M 1111267 IC50 = 9.7 nM T02562 C7XM3U 1129243 IC50 = 54500 nM T02562 C9X3AF 1144445 IC50 = 3600 nM T02562 CEY8N7 1144449 IC50 = 700 nM T02562 C4WK8N 1147431 IC50 = 9200 nM T02562 CO1C4E 1151293 IC50 = 7500 nM T02562 CL3SK9 1206529 IC50 = 800 nM T02562 CJ0TX2 1232170 IC50 = 160000 nM T02562 CWA0B4 1240120 IC50 = 2300 nM T02562 CUWO38 1355190 IC50 = 1100 nM T02562 CILN42 1356792 IC50 = 3800 nM T02562 CJQ0B9 1594408 IC50 = 1.8 nM T02562 C50DMX 1719649 IC50 = 1700 nM T02562 CFE92U 1723288 IC50 = 2800 nM T02562 C24LCO 1797625 IC50 = 4400 nM T02562 CBY96N 1809082 IC50 = 100 nM T02562 CM3X2R 1822643 IC50 = 3600 nM T02562 CP4RT3 2190043 IC50 = 710 nM T02562 C7ECR6 2200735 IC50 = 240 nM T02562 C38UEP 2205605 IC50 = 100 nM T02562 C45LQX 2841002 IC50 = 16900 nM T02562 CDQ97L 2883254 IC50 = 5700 nM T02562 C60OPF 2883266 IC50 = 8800 nM T02562 C5G9LJ 2895777 IC50 = 1600 nM T02562 CQKW21 2972602 IC50 = 2 nM T02562 CE6JY3 2991119 IC50 = 32500 nM T02562 CWH14B 3002003 IC50 = 370 nM T02562 CVU5O1 3108985 IC50 = 7900 nM T02562 C31ZNO 3109454 IC50 = 10 nM T02562 CGR7T8 3126444 IC50 > 100000 nM T02562 CEQ2Z5 3151671 IC50 = 9600 nM T02562 C78RPF 3165998 IC50 = 19400 nM T02562 CB4IF8 3166828 IC50 = 930 nM T02562 CB4E8U 3170441 IC50 = 13800 nM T02562 CF6CV0 3188168 IC50 = 180 nM T02562 C3GM2V 3188196 IC50 = 360 nM T02562 CV56AO 3188216 IC50 = 220 nM T02562 C4ORF2 3188301 IC50 = 180 nM T02562 C5B6XO 3188315 IC50 = 130 nM T02562 C6GR1D 3201860 IC50 = 210 nM T02562 C3QYZ8 3316916 IC50 = 3700 nM T02562 CF4U2J 3975154 IC50 = 1800 nM T02562 CZ21OV 4426033 IC50 = 200 nM T02562 CJ0D1G 4589007 IC50 = 7700 nM T02562 CDP47N 4637714 IC50 = 12600 nM T02562 C4E3MH 4645817 IC50 = 23600 nM T02562 CK98IS 4690153 IC50 > 50000 nM T02562 C6H2SP 5185168 IC50 = 2600 nM T02562 C4SQ5B 5296590 IC50 = 1000 nM T02562 CV8L7N 5342141 IC50 = 2 nM T02562 C13OPQ 5352088 IC50 = 300 nM T02562 C7MP4R 5910939 IC50 = 4600 nM T02562 C4O0VE 5957759 IC50 = 1900 nM T02562 C0BY6F 6261723 IC50 = 11000 nM T02562 CAFX48 6402421 IC50 = 2500 nM T02562 C32TMK 6403001 IC50 = 5000 nM T02562 CWC8D2 6406804 IC50 = 45400 nM T02562 CT38JI 6408881 IC50 = 17800 nM T02562 CF83PE 6408905 IC50 = 290 nM T02562 C60NWA 6409077 IC50 = 480 nM T02562 CIAV08 6409184 IC50 = 50800 nM T02562 C4WYA1 6411927 IC50 = 13900 nM T02562 CRUQ02 6414877 IC50 = 500 nM T02562 C9JBH5 6415933 IC50 = 2100 nM T02562 C05CNL 6418564 IC50 = 32900 nM T02562 CQO9T1 6440631 IC50 = 13000 nM T02562 C0SN3Z 6917852 IC50 = 45000 nM T02562 CRTU70 8075068 IC50 = 1500 nM T02562 C4W2JR 9498257 IC50 = 120000 nM T02562 CGR29L 9525248 IC50 = 4 nM T02562 CIAR14 9532977 IC50 = 6.5 nM T02562 CD17IV 9654525 IC50 = 66000 nM T02562 C9XS8E 9662597 IC50 = 100 nM T02562 C8TEO4 10071695 IC50 = 1800 nM T02562 CKS74T 10132240 IC50 = 4600 nM T02562 CJ4ZO7 10355545 IC50 = 7400 nM T02562 CM7X8L 10449221 IC50 = 20 nM T02562 CU28FC 10522757 IC50 = 670 nM T02562 CL6T2N 10638828 IC50 = 9300 nM T02562 C23VDE 10999992 IC50 = 19500 nM T02562 C1XF8A 11385862 IC50 = 2100 nM T02562 CP2ID5 11386458 IC50 = 3000 nM T02562 C5L7IW 11510178 IC50 = 2580 nM T02562 C2XQI7 11526708 IC50 = 23 nM T02562 CYKR80 11545682 IC50 = 600 nM T02562 CXS9A3 11562170 IC50 = 1 nM T02562 CZ08BT 11576785 IC50 = 1 nM T02562 C5HG9T 11583832 IC50 = 1 nM T02562 C3Z7IS 11590429 IC50 = 60 nM T02562 CO8LJ4 11592681 IC50 = 490 nM T02562 CM3D5X 11669713 IC50 = 9 nM T02562 CE4S2G 11687311 IC50 > 10000 nM T02562 CR06AO 11692277 IC50 = 2 nM T02562 CX91IU 11698651 IC50 = 57 nM T02562 C45NBF 11705274 IC50 = 13 nM T02562 CKG9V6 11707099 IC50 = 390 nM T02562 CQT67H 11712400 IC50 = 0.7 nM T02562 CN7TS9 11777067 IC50 = 7100 nM T02562 CVT0F8 11808877 IC50 = 3500 nM T02562 CWF6I8 11841193 IC50 = 20000 nM T02562 CJO9Z6 11978569 IC50 = 5100 nM T02562 CN8RP5 12306720 IC50 = 400 nM T02562 CCZL29 12315005 IC50 > 10000 nM T02562 CTQ31G 12658321 IC50 = 6400 nM T02562 CPVK13 12997791 IC50 > 10000 nM T02562 CX54UL 12997794 IC50 > 10000 nM T02562 C3X7TM 12997796 IC50 = 2500 nM T02562 C5LH9S 14213209 IC50 > 50000 nM T02562 CZUI98 14213211 IC50 = 42000 nM T02562 C0GLC7 14213215 IC50 = 13500 nM T02562 CIT35C 14213224 IC50 > 50000 nM T02562 C9MNS6 14471387 IC50 = 3600 nM T02562 CWM83A 14845590 IC50 > 10000 nM T02562 CVQ03M 14855811 IC50 = 1800 nM T02562 C8SY2C 14855860 IC50 = 7200 nM T02562 CNV7D6 15110283 IC50 = 11300 nM T02562 C13DIN 15940274 IC50 = 60 nM T02562 C40KNM 16046096 IC50 = 1300 nM T02562 C6P7DY 16046097 IC50 = 1100 nM T02562 C1WJ2D 16070041 IC50 = 1 nM T02562 C3Q4EG 16112833 IC50 = 0.9 nM T02562 CI0E7J 16220835 IC50 > 10000 nM T02562 CL0Y9O 16727118 IC50 = 3940 nM T02562 C6Y2BV 16730199 IC50 = 2 nM T02562 CB38HP 16730202 IC50 = 3 nM T02562 CUJH07 16730353 IC50 = 1 nM T02562 C4N1EY 16733250 IC50 = 60 nM T02562 CKE41X 16753429 IC50 = 2600 nM T02562 CXN0W2 21581528 IC50 = 8500 nM T02562 CFT46C 22574175 IC50 = 560 nM T02562 CC8JB3 24721570 IC50 = 900 nM T02562 C59FKG 24860777 IC50 = 36 nM T02562 C1LE0A 24860912 IC50 = 2 nM T02562 C9XJ1Q 24861146 IC50 = 6 nM T02562 C13QJO 24861205 IC50 = 7 nM T02562 C1M8ZP 24861261 IC50 = 4 nM T02562 CJU54K 24861311 IC50 = 45 nM T02562 C3C2ME 24861314 IC50 = 7 nM T02562 CX4BC5 24861472 IC50 = 1000 nM T02562 CF3B5Y 24861474 IC50 = 1 nM T02562 C2F9XY 24971276 IC50 = 5600 nM T02562 C7Y4GR 25058073 IC50 = 600 nM T02562 CXH48N 25058075 IC50 = 300 nM T02562 C6RZC2 25147690 IC50 = 650 nM T02562 C0PAE1 25179516 IC50 > 10000 nM T02562 C5RBW3 25179712 IC50 = 1700 nM T02562 CL3Q7B 25179713 IC50 = 2100 nM T02562 C54DIT 25179907 IC50 = 1200 nM T02562 C9GB6J 25179909 IC50 = 1600 nM T02562 CC9N3E 25179911 IC50 = 2100 nM T02562 CUTK18 25179912 IC50 = 1600 nM T02562 C1T2HP 25205185 IC50 = 10200 nM T02562 CFY5T4 25608033 IC50 = 640 nM T02562 CYZ6B0 26389403 IC50 > 50000 nM T02562 CA89YP 41160317 IC50 > 100000 nM T02562 CH0G2S 42610408 IC50 = 10 nM T02562 CY4CX1 44157329 IC50 = 1600 nM T02562 CV7CF8 44157483 IC50 = 960 nM T02562 C97ING 44157555 IC50 = 3400 nM T02562 CU5IN7 44157725 IC50 = 600 nM T02562 CUGY90 44157824 IC50 = 3400 nM T02562 CYIX03 44157825 IC50 = 500 nM T02562 CH59LF 44157826 IC50 = 200 nM T02562 CTA48Z 44157827 IC50 = 600 nM T02562 CY29SV 44157829 IC50 = 6010 nM T02562 CLP20K 44157929 IC50 = 1700 nM T02562 CPEF24 44221149 IC50 = 4500 nM T02562 C6EW9A 44221151 IC50 = 3900 nM T02562 CHY6D9 44221548 IC50 = 5900 nM T02562 C2Y9IT 44221753 IC50 = 4800 nM T02562 CSBW72 44221754 IC50 = 2100 nM T02562 C98GDR 44249905 IC50 = 4200 nM T02562 C9O7QC 44389542 IC50 = 6700 nM T02562 CH2V4K 44389592 IC50 = 3200 nM T02562 CZ4P1W 44389720 IC50 = 900 nM T02562 CUW8S1 44390083 IC50 = 260 nM T02562 C6XN8F 44390610 IC50 = 16 nM T02562 CI3BM4 44390722 IC50 = 3 nM T02562 C69GNE 44390943 IC50 = 4 nM T02562 C75XZW 44469536 IC50 = 900 nM T02562 CU05BN 44538798 IC50 = 2800 nM T02562 CP4AV0 44585939 IC50 = 60 nM T02562 C21DRI 44585940 IC50 = 70 nM T02562 CLP0D9 44587062 IC50 = 1000 nM T02562 CJH3U6 45102382 IC50 = 2000 nM T02562 CAXW02 45110606 IC50 = 2100 nM T02562 CL9MY2 45112300 IC50 = 30 nM T02562 CSLZ04 45267718 IC50 > 10000 nM T02562 C0R8MQ 45267726 IC50 = 4100 nM T02562 C8AXK3 45268597 IC50 = 2000 nM T02562 C6CEX5 45268605 IC50 > 10000 nM T02562 C0F7RJ 45268611 IC50 = 7100 nM T02562 C1EIF5 45269442 IC50 > 10000 nM T02562 CU91HN 45269452 IC50 = 2200 nM T02562 C74OGR 45269453 IC50 > 10000 nM T02562 C59HVY 45269638 IC50 = 6200 nM T02562 C4X8NT 45270286 IC50 = 2700 nM T02562 CJC3M7 45270291 IC50 > 10000 nM T02562 CTX61C 45271105 IC50 = 4600 nM T02562 C5U8HX 45271112 IC50 = 1700 nM T02562 CR1QU8 45271974 IC50 > 10000 nM T02562 CN4ET7 45271983 IC50 = 8800 nM T02562 CH92UP 45271992 IC50 > 10000 nM T02562 C42QTW 45272810 IC50 = 9300 nM T02562 CVU12R 45272820 IC50 = 2200 nM T02562 COP75F 45273770 IC50 = 2900 nM T02562 CQ4GE9 45273780 IC50 > 10000 nM T02562 CC24IR 45276264 IC50 = 930 nM T02562 C7TI8O 45487784 IC50 = 11 nM T02562 CW2YP7 45487785 IC50 = 1 nM T02562 C16OEZ 45487788 IC50 = 5000 nM T02562 CL09DY 45487795 IC50 = 25 nM T02562 C1N2LK 45487799 IC50 = 1 nM T02562 CU23OF 45487804 IC50 = 8 nM T02562 CTD07E 45487806 IC50 = 8 nM T02562 CM04KU 45487816 IC50 = 122 nM T02562 CN36KB 45487834 IC50 = 710 nM T02562 CFHN68 45487835 IC50 = 4 nM T02562 CJ1UN6 45487836 IC50 = 0.4 nM T02562 CM71IC 45487840 IC50 = 3 nM T02562 CZL7E6 46189367 IC50 = 1100 nM T02562 C6GK7O 46213655 IC50 = 2 nM T02562 CH52BL 46227442 IC50 = 3100 nM T02562 C1XDO6 46834705 IC50 = 6970 nM T02562 C2RTO6 46837638 IC50 = 7300 nM T02562 CM2K0V 46837639 IC50 = 2000 nM T02562 CRY5B0 46837640 IC50 = 1200 nM T02562 CY85OT 46837641 IC50 = 3800 nM T02562 C2OP7F 46837642 IC50 = 2200 nM T02562 CHJD18 46837643 IC50 = 900 nM T02562 CIH0K4 46837775 IC50 = 900 nM T02562 CP8OA1 46837776 IC50 > 10000 nM T02562 CV5ZO3 46837777 IC50 = 1900 nM T02562 CWFQ46 46837778 IC50 > 10000 nM T02562 CD37LB 46837779 IC50 = 3700 nM T02562 CEPL58 46837915 IC50 = 5900 nM T02562 C89OMP 46837916 IC50 = 6500 nM T02562 C5YJS7 46837917 IC50 > 10000 nM T02562 CM3H5J 46837918 IC50 = 2400 nM T02562 CKDW89 46837919 IC50 > 10000 nM T02562 CD5UE3 46837920 IC50 = 9600 nM T02562 C4S6ID 46838058 IC50 > 10000 nM T02562 CET7R4 46866190 IC50 = 5700 nM T02562 CRQ29W 46880352 IC50 = 190 nM T02562 CN62CQ 46880353 IC50 = 5760 nM T02562 C0E3BU 46880390 IC50 = 29600 nM T02562 C30YCD 46881260 IC50 = 2000 nM T02562 C08GUA 46885478 IC50 = 1900 nM T02562 CSU0B6 46885553 IC50 = 5100 nM T02562 CP3EV2 46885590 IC50 = 6100 nM T02562 C9TCN2 46908258 IC50 = 0.1 nM T02562 C5QM3O 46908736 IC50 = 3 nM T02562 C4UI9E 49839479 IC50 = 1 nM T02562 CSKZ81 50997363 IC50 = 25 nM T02562 CH82SZ 51000500 IC50 = 47 nM T02562 C4R8ZK 51136453 IC50 = 820 nM T02562 CZD5R6 51346789 IC50 = 940 nM T02562 C84JTI 51346790 IC50 = 900 nM T02562 CJP9O3 51346855 IC50 = 330 nM T02562 C4MH8K 51355427 IC50 < 3200 nM T02562 CIT7W2 51534485 IC50 = 7900 nM T02562 CEX0K1 51976272 IC50 = 1300 nM T02562 CTO0P3 52919086 IC50 = 2 nM T02562 CAZ68S 52941010 IC50 = 3700 nM T02562 CLS0R8 52942224 IC50 > 30000 nM T02562 CD4S5X 52943616 IC50 = 1400 nM T02562 C8GQ6H 52943812 IC50 = 4 nM T02562 CB08CT 52945864 IC50 = 1300 nM T02562 CCB50A 52946331 IC50 = 940 nM T02562 C58DMR 53252516 IC50 = 3 nM T02562 C6G7ZT 53317142 IC50 = 880 nM T02562 CJ34IB 53317510 IC50 = 31 nM T02562 C80GXT 53317600 IC50 = 3500 nM T02562 CGNT20 53317601 IC50 = 1100 nM T02562 C6J4DK 53317602 IC50 = 910 nM T02562 CF27US 53317603 IC50 = 150 nM T02562 C08TYZ 53317604 IC50 = 480 nM T02562 C7WD8P 53317700 IC50 = 2 nM T02562 CHN76K 53318433 IC50 = 1600 nM T02562 CW61TX 53318885 IC50 = 660 nM T02562 C8XAT4 53318886 IC50 = 580 nM T02562 C9E4LM 53318887 IC50 = 18 nM T02562 C1PCF3 53318888 IC50 = 32 nM T02562 CFP6I8 53319766 IC50 = 940 nM T02562 C71WEJ 53320101 IC50 = 46 nM T02562 C7KDY2 53320202 IC50 = 1800 nM T02562 CGA52E 53320203 IC50 = 8 nM T02562 CI70QH 53320204 IC50 = 48 nM T02562 CZ2UX6 53320205 IC50 = 7900 nM T02562 C7KZ8M 53320206 IC50 = 43 nM T02562 CG49YR 53320386 IC50 > 10000 nM T02562 C89KRP 53321057 IC50 = 1550 nM T02562 C6FIA3 53321130 IC50 = 3000 nM T02562 CB5PC9 53321521 IC50 = 150 nM T02562 C31BJP 53321522 IC50 = 18 nM T02562 CEO2R3 53321617 IC50 = 3 nM T02562 C5Q1XK 53322727 IC50 = 4500 nM T02562 CDU1Q2 53322728 IC50 = 4200 nM T02562 CG37XR 53322832 IC50 = 1700 nM T02562 CWLZ92 53322849 IC50 = 990 nM T02562 CJI8N3 53324175 IC50 = 190 nM T02562 CGS68Y 53325027 IC50 = 1500 nM T02562 CTP62K 53325474 IC50 = 22 nM T02562 CC0KS4 53325475 IC50 = 9 nM T02562 C30EUD 53325476 IC50 = 1 nM T02562 CCUN93 53325477 IC50 > 10000 nM T02562 CH8YK2 53325478 IC50 = 1600 nM T02562 C2WPA0 53325579 IC50 = 1300 nM T02562 C4J5DH 53326328 IC50 = 1900 nM T02562 C6JUK8 53326329 IC50 = 1450 nM T02562 CN48MT 53326634 IC50 = 9700 nM T02562 C8S9ND 53326734 IC50 = 13 nM T02562 CO1G8Y 53326735 IC50 = 3 nM T02562 CP1A7T 53326736 IC50 = 12 nM T02562 CC7KT6 53363130 IC50 = 4600 nM T02562 CF5U2R 53363131 IC50 = 3400 nM T02562 CSC3V7 53363132 IC50 = 2400 nM T02562 CH2DO7 53363133 IC50 = 2800 nM T02562 CPD82G 53363134 IC50 = 3900 nM T02562 CI4D2P 53363220 IC50 = 2700 nM T02562 C2O8FZ 53363221 IC50 > 10000 nM T02562 CX7I2Y 53363222 IC50 = 2400 nM T02562 C5H6YT 53363223 IC50 = 1100 nM T02562 C1WB4D 53363224 IC50 = 1500 nM T02562 CUI04W 53363313 IC50 = 3500 nM T02562 CY3OX0 53363314 IC50 > 10000 nM T02562 C8G0LH 53363315 IC50 > 10000 nM T02562 CB34MJ 53363401 IC50 = 3400 nM T02562 C7WAJ2 53439651 IC50 = 10000 nM T02562 C1EFU6 53483951 IC50 = 5300 nM T02562 C9LMW2 54583638 IC50 > 10000 nM T02562 CR1DH4 54585240 IC50 = 5100 nM T02562 C6LTB2 54585561 IC50 = 9400 nM T02562 C7NHS0 54586204 IC50 = 2600 nM T02562 CSRV19 54586205 IC50 = 3900 nM T02562 C2IB5H 54682566 IC50 = 400 nM T02562 C87GPY 54728405 IC50 = 110 nM T02562 C0X6ZQ 54728406 IC50 = 290 nM T02562 CC1Y9K 54728407 IC50 = 530 nM T02562 CROP60 54728408 IC50 = 150 nM T02562 C76ETO 54728409 IC50 = 1140 nM T02562 CR0E7X 54728410 IC50 = 2160 nM T02562 C1ZR3C 54728411 IC50 = 3440 nM T02562 CRNV32 54728412 IC50 = 3960 nM T02562 CAP19Z 54728413 IC50 = 3130 nM T02562 C3IXM4 54728414 IC50 = 16 nM T02562 C0NTK4 54728415 IC50 < 920 nM T02562 CT3PE0 54728416 IC50 < 760 nM T02562 CPD72H 54728417 IC50 = 1000 nM T02562 CW6ZG1 54728418 IC50 = 32200 nM T02562 CFT90G 54728419 IC50 = 160 nM T02562 C08YMI 54728420 IC50 = 12700 nM T02562 CXH87Q 54728421 IC50 = 65600 nM T02562 CMW56Z 54728422 IC50 = 11700 nM T02562 C3XW4R 54728423 IC50 = 1290 nM T02562 C7DY8K 54728424 IC50 = 1450 nM T02562 CZB47W 54728425 IC50 = 3050 nM T02562 CJ0XK5 54728426 IC50 = 180 nM T02562 CI4TA5 54728427 IC50 = 280 nM T02562 C14MSR 54728428 IC50 < 70 nM T02562 CG9ZC5 54728429 IC50 < 26 nM T02562 CHEA98 54754344 IC50 = 3500 nM T02562 C79DVG 56589615 IC50 = 4.1 nM T02562 CD7TI0 56649439 IC50 = 65 nM T02562 C0Y4OK 56649440 IC50 = 88 nM T02562 CY3G8F 56834936 IC50 = 9.1 nM T02562 CEN59P 56837793 IC50 = 4 nM T02562 CK6Y7X 56955459 IC50 = 4850 nM T02562 C6BC7L 56968260 IC50 = 12 nM T02562 CPQB48 56968267 IC50 = 3.7 nM T02562 C14USR 56968481 IC50 = 5.8 nM T02562 C1PF9M 56968482 IC50 = 26 nM T02562 C4UZS3 56968711 IC50 = 25 nM T02562 C2T0XE 56968925 IC50 = 7.8 nM T02562 CJI80B 56968927 IC50 = 6.5 nM T02562 C54WCS 56968928 IC50 = 13 nM T02562 CFJX09 56969153 IC50 = 6.7 nM T02562 CP39FD 56969373 IC50 = 2.3 nM T02562 C5W9TL 56969375 IC50 = 11 nM T02562 CGH1Q3 56969599 IC50 = 13 nM T02562 C56ZNH 56969601 IC50 = 23 nM T02562 CDBX04 56969811 IC50 = 4.9 nM T02562 CJD1S3 56970017 IC50 = 6.4 nM T02562 CY0X2A 56970021 IC50 = 47 nM T02562 C7OHF1 56970442 IC50 = 4.1 nM T02562 C1AV7C 56970444 IC50 = 14 nM T02562 CQ9J8H 56970445 IC50 = 30 nM T02562 C2A0UN 56970656 IC50 = 6.1 nM T02562 C3OF0J 56970893 IC50 = 29 nM T02562 CL14JA 56971113 IC50 = 3.6 nM T02562 CX3AR0 56971116 IC50 = 3.1 nM T02562 CWBN09 56971351 IC50 = 3.2 nM T02562 CJ3SN0 56971576 IC50 = 9.4 nM T02562 CT7YS0 57326556 IC50 = 800 nM T02562 C7U9TI 57326557 IC50 = 1000 nM T02562 CI07KF 57328416 IC50 = 140 nM T02562 C9CKB0 57328574 IC50 = 600 nM T02562 CX37LB 57382526 IC50 = 0.744 nM T02562 C1NDL3 57390737 IC50 = 506 nM T02562 CT7DN8 57392544 IC50 > 10000 nM T02562 CE8AC5 57392545 IC50 = 330 nM T02562 C9UE5B 57394266 IC50 > 10000 nM T02562 CTU5A8 57394267 IC50 = 4620 nM T02562 C5F9BK 57394268 IC50 = 687 nM T02562 CORQ69 57394269 IC50 = 6264 nM T02562 CJ25ZL 57394270 IC50 = 172 nM T02562 CO4M5L 57396016 IC50 = 1000 nM T02562 C9JI5R 57397813 IC50 = 1490 nM T02562 CP48IT 57397814 IC50 = 306 nM T02562 CWCB25 57397815 IC50 = 108 nM T02562 C6ARY7 57397881 IC50 = 9500 nM T02562 CES91N 57399484 IC50 = 395 nM T02562 CT2VC7 57399485 IC50 = 669 nM T02562 CTGX92 57401247 IC50 = 62 nM T02562 CX39GR 57402990 IC50 = 251 nM T02562 CH39OB 57402991 IC50 = 859 nM T02562 C1EF8K 57412312 IC50 = 370 nM T02562 CTPW84 57412314 IC50 = 260 nM T02562 C5HQ1A 57700184 IC50 = 340 nM T02562 CMR61U 59581717 IC50 > 2000 nM T02562 CX6QY4 60148597 IC50 = 24.76 nM T02562 CTQM50 60148675 IC50 = 1400 nM T02562 CHI25V 60163714 IC50 = 61.81 nM T02562 C6LO8K 60163716 IC50 = 796.7 nM T02562 CW73KB 60163802 IC50 = 640.8 nM T02562 CF7P6Z 60163882 IC50 = 9.3 nM T02562 CO73IK 60163884 IC50 = 39.16 nM T02562 CKP89Y 60163885 IC50 = 28.2 nM T02562 CM49CX 60163965 IC50 = 29.31 nM T02562 CH5S3B 60163967 IC50 = 15.61 nM T02562 CYL49R 60163968 IC50 = 29.65 nM T02562 CL71GR 60163969 IC50 = 838.7 nM T02562 C0MHI8 60164046 IC50 = 464.8 nM T02562 CI39NC 60164047 IC50 = 12.28 nM T02562 C4TIW9 60164359 IC50 = 33.06 nM T02562 CRJN30 60164486 IC50 = 169.7 nM T02562 C4SL0P 60164591 IC50 = 3.89 nM T02562 CFHU69 60164592 IC50 = 15.9 nM T02562 CWK28F 60164593 IC50 = 12.65 nM T02562 CD4P5H 60164702 IC50 = 407 nM T02562 CU24XS 60164916 IC50 = 252.2 nM T02562 CMG87U 60165011 IC50 = 325.2 nM T02562 C9ARQ4 60165012 IC50 = 709.5 nM T02562 C0AN9J 60172692 IC50 = 20 nM T02562 C9YE0M 60200527 IC50 = 4200 nM T02562 CLM07N 60200528 IC50 = 1900 nM T02562 C01PGH 60200529 IC50 = 2700 nM T02562 CJA2K5 66560429 IC50 = 900 nM T02562 CGC85K 66560430 IC50 = 5600 nM T02562 CHW2I8 66571763 IC50 > 10000 nM T02562 C5K2CY 66571764 IC50 > 10000 nM T02562 CY4X5D 66571765 IC50 > 10000 nM T02562 C0G1LM 66571766 IC50 > 10000 nM T02562 CKT32E 66571767 IC50 > 10000 nM T02562 C1P3RA 66571860 IC50 = 1200 nM T02562 CTW74V 66571861 IC50 = 5500 nM T02562 CES4Y3 66571862 IC50 > 10000 nM T02562 CF96OW 66571863 IC50 > 10000 nM T02562 C5H2ZY 66571963 IC50 = 680 nM T02562 C7YPV3 66571964 IC50 = 1000 nM T02562 CX04YA 66571965 IC50 > 10000 nM T02562 C8DY7B 66573411 IC50 > 10000 nM T02562 C0B7CK 66573412 IC50 > 10000 nM T02562 C5I3XH 66573413 IC50 > 10000 nM T02562 CL97EK 67033699 IC50 = 90 nM T02562 COAP48 67502417 IC50 = 3.9 nM T02562 CI93YX 67502703 IC50 = 32 nM T02562 COE02J 67502724 IC50 = 17 nM T02562 CY7WA5 67503084 IC50 = 58 nM T02562 CVK58R 67503100 IC50 = 10 nM T02562 C57MFJ 67503146 IC50 = 22 nM T02562 C8B2VR 67503231 IC50 = 2.8 nM T02562 CL1P9V 67503311 IC50 = 11 nM T02562 CS3W0I 67503321 IC50 = 4 nM T02562 C0JQ1B 67503326 IC50 = 157 nM T02562 CT27ZB 67503330 IC50 = 4.9 nM T02562 CQG1R2 67503337 IC50 = 6.3 nM T02562 CDK15T 67503464 IC50 = 14 nM T02562 C8YT7R 67503471 IC50 = 154.2 nM T02562 C4VK8P 67503476 IC50 = 405 nM T02562 CO5I3S 67503518 IC50 = 3.3 nM T02562 CHO02W 67503542 IC50 = 5.4 nM T02562 C5YV4F 67503554 IC50 = 82 nM T02562 C0SX7Q 67503727 IC50 = 10 nM T02562 C8VUX5 67503753 IC50 = 4.1 nM T02562 CEN36P 67503787 IC50 = 4.6 nM T02562 CT50HR 67503968 IC50 = 10 nM T02562 CL3RX8 67504002 IC50 = 3.7 nM T02562 C92RKJ 67504009 IC50 = 47 nM T02562 CSP30R 67504030 IC50 = 9.7 nM T02562 CPYG57 67504351 IC50 = 39 nM T02562 CTE6X3 67504414 IC50 = 3.5 nM T02562 C39OSM 67970587 IC50 = 2.32 nM T02562 C8K0EX 67970734 IC50 = 0.792 nM T02562 C2VN0R 67970797 IC50 = 3.15 nM T02562 CH4K6P 67970801 IC50 = 3.67 nM T02562 CE7JZ8 67970931 IC50 = 1.08 nM T02562 C9H0RE 67970984 IC50 = 3.11 nM T02562 C5Y4HQ 67971014 IC50 = 0.385 nM T02562 CDX5W8 67971063 IC50 = 1.43 nM T02562 CM90KH 67971414 IC50 = 0.198 nM T02562 C5G4VJ 67990975 IC50 = 1.12 nM T02562 C6B9TW 68282786 IC50 = 81.28 nM T02562 C5TQ7W 68282799 IC50 = 64.68 nM T02562 C9J0QW 68282901 IC50 = 320 nM T02562 CF9LC8 68283167 IC50 = 83.02 nM T02562 C5PG7J 68283220 IC50 = 12.72 nM T02562 C8T9DW 68283231 IC50 = 35.55 nM T02562 C6M4KG 68283242 IC50 = 11.22 nM T02562 C8L5QA 68283250 IC50 = 19.85 nM T02562 CF3A9J 68283276 IC50 = 11.77 nM T02562 CV0NJ9 68283277 IC50 = 38.24 nM T02562 C0I1SJ 68352348 IC50 = 191.4 nM T02562 CIH2U0 71059686 IC50 = 720 nM T02562 CB8E1W 71059857 IC50 = 10.3 nM T02562 C3CD4P 71059962 IC50 < 3 nM T02562 C2COY0 71296422 IC50 = 2100 nM T02562 CS3RK5 71451782 IC50 = 1800 nM T02562 CUA81S 71451783 IC50 = 2800 nM T02562 C53HRS 71451785 IC50 = 800 nM T02562 C7HVK4 71453597 IC50 = 1700 nM T02562 CV8N3Q 71453598 IC50 = 2500 nM T02562 CWYG47 71455331 IC50 = 160 nM T02562 CFJC03 71455332 IC50 = 180 nM T02562 CB34ZQ 71455333 IC50 = 350 nM T02562 C4QE3U 71455826 IC50 = 1700 nM T02562 CRS19Y 71457107 IC50 = 1750 nM T02562 CB1Q5R 71458972 IC50 = 400 nM T02562 CL16CK 71458973 IC50 = 3400 nM T02562 CPVC31 71460125 IC50 = 39500 nM T02562 CH3YD6 71460772 IC50 = 200 nM T02562 C9HK3Z 71462499 IC50 = 5900 nM T02562 CCDU47 71462500 IC50 = 2300 nM T02562 CF6M7N 71462978 IC50 = 900 nM T02562 CJ87CO 71515675 IC50 = 157 nM T02562 CN2H3W 71516251 IC50 = 3 nM T02562 CVUQ15 71517338 IC50 = 6900 nM T02562 CSY9N3 71517339 IC50 = 10300 nM T02562 C6B8PZ 71517340 IC50 = 9700 nM T02562 CWP01A 71517341 IC50 = 4100 nM T02562 C1VS8N 71517501 IC50 = 4000 nM T02562 CKZ25C 71517502 IC50 = 1100 nM T02562 C9UH5F 71517503 IC50 = 4200 nM T02562 CB37TY 71517504 IC50 = 3800 nM T02562 CKPT54 71517505 IC50 = 3300 nM T02562 CT0O7G 71517506 IC50 = 4400 nM T02562 CG68NS 71517507 IC50 = 12900 nM T02562 C1S4GA 71517673 IC50 = 6300 nM T02562 C9YCI3 71520910 IC50 = 850 nM T02562 C27KUX 71520911 IC50 > 10000 nM T02562 C84RCV 71520912 IC50 > 10000 nM T02562 CQI76N 71520913 IC50 > 10000 nM T02562 CF2R6B 71520914 IC50 = 12900 nM T02562 CTF2P5 71521012 IC50 > 30000 nM T02562 CZ7MW2 71521013 IC50 = 3010 nM T02562 C37IJV 71521014 IC50 = 1680 nM T02562 CLN02O 71521015 IC50 = 821 nM T02562 C8NH5T 71521016 IC50 = 242 nM T02562 CV6P4F 71521017 IC50 = 291 nM T02562 C8I7RK 71521018 IC50 = 7180 nM T02562 C0NSO7 71521120 IC50 = 8150 nM T02562 C3J4BK 71521121 IC50 = 826 nM T02562 C45ZGP 71521122 IC50 = 176 nM T02562 CPF2G8 71521123 IC50 = 220 nM T02562 CC0KA9 71521124 IC50 = 785 nM T02562 CN0OF2 71521223 IC50 = 3200 nM T02562 CT2OL8 71521224 IC50 = 43.1 nM T02562 CFV62N 71521225 IC50 = 34 nM T02562 CEJU20 71521226 IC50 = 82 nM T02562 C2H8SM 71521227 IC50 = 40 nM T02562 CJ7NY0 71532255 IC50 = 0.1 nM T02562 C91UFR 71552025 IC50 = 33 nM T02562 CL8D5U 71552026 IC50 = 336 nM T02562 CL0JP5 71552027 IC50 = 3 nM T02562 C1GS4A 71552028 IC50 = 3 nM T02562 CW6L9R 71552029 IC50 = 3 nM T02562 C0WYL5 71552106 IC50 = 2 nM T02562 C57WJZ 71552270 IC50 = 72 nM T02562 C9PZJ7 71552271 IC50 = 600 nM T02562 CAM6W7 71552272 IC50 = 610 nM T02562 CCB36A 71552359 IC50 = 1900 nM T02562 CH54EK 71552360 IC50 = 34 nM T02562 C65EAT 71552361 IC50 = 1400 nM T02562 CE6SC4 71552362 IC50 = 8.3 nM T02562 CE9K6I 71552363 IC50 = 16 nM T02562 CX0M9Z 71552364 IC50 = 250 nM T02562 CD16KP 71553158 IC50 = 6750 nM T02562 CASN52 71553159 IC50 = 47 nM T02562 CZF75T 71553160 IC50 = 9800 nM T02562 C08YCU 71553161 IC50 > 33000 nM T02562 C0ZPC6 71553162 IC50 > 33000 nM T02562 CLC9V7 71553245 IC50 = 88 nM T02562 CRX0W1 71553246 IC50 = 25 nM T02562 CD5FZ3 71553247 IC50 = 20 nM T02562 C1N9TO 71553248 IC50 = 6 nM T02562 CQRS94 71553249 IC50 = 761 nM T02562 CPO6A0 71553250 IC50 = 16 nM T02562 CSBO80 71569485 IC50 = 5 nM T02562 CMVT07 71570309 IC50 < 50 nM T02562 C7R5EZ 71571581 IC50 = 8700 nM T02562 CWOU26 71583753 IC50 = 9810 nM T02562 CK29IY 71583754 IC50 > 10000 nM T02562 CVBN29 71583755 IC50 = 85 nM T02562 CHR26Q 71583756 IC50 > 10000 nM T02562 CSD8W1 71583757 IC50 > 10000 nM T02562 CQO29N 71583758 IC50 = 106 nM T02562 CN20LT 71583759 IC50 = 226 nM T02562 C6DCO1 71583872 IC50 = 1068 nM T02562 C3V9AM 71583873 IC50 = 631 nM T02562 C43RLU 71583874 IC50 = 387 nM T02562 C16WBP 71583875 IC50 = 31 nM T02562 CB4K9V 71583876 IC50 = 59 nM T02562 C10BDU 71583877 IC50 = 83 nM T02562 C61RYH 71659356 IC50 = 891 nM T02562 CVDB58 71659357 IC50 = 27 nM T02562 C28EIT 71659358 IC50 = 198 nM T02562 C8DF4B 71659489 IC50 = 434 nM T02562 C7Y0RM 71659490 IC50 = 241 nM T02562 CKR47S 71659491 IC50 = 98 nM T02562 CAQ2V1 71659492 IC50 = 17 nM T02562 CJX32Y 71659493 IC50 = 53 nM T02562 C05JLG 71659494 IC50 = 70 nM T02562 COS6Q5 71659610 IC50 = 17 nM T02562 CNVI07 71659611 IC50 = 21 nM T02562 CUF06Z 71659612 IC50 = 7.9 nM T02562 CT9KZ0 71659613 IC50 = 32 nM T02562 CZFU74 71659614 IC50 = 21 nM T02562 CC3L1Y 71659615 IC50 = 22 nM T02562 CF1HA9 71659751 IC50 = 908 nM T02562 CF8DV2 71659752 IC50 = 1128 nM T02562 CMA4N0 71659753 IC50 = 9.9 nM T02562 CFBA41 71659754 IC50 = 4.5 nM T02562 CR58TZ 71659755 IC50 = 8.3 nM T02562 CVE91N 71659756 IC50 = 4.3 nM T02562 CH4VF0 71659894 IC50 = 2.5 nM T02562 C53AOG 71659895 IC50 = 3.3 nM T02562 C9WC2J 71659896 IC50 = 12 nM T02562 CTBX46 71659897 IC50 = 12 nM T02562 CW0Y5N 71659898 IC50 = 10 nM T02562 CGE1V8 71717945 IC50 = 23300 nM T02562 CG80HX 71718897 IC50 = 3100 nM T02562 CA5UT3 71719199 IC50 = 1200 nM T02562 C7STX5 71719487 IC50 = 54 nM T02562 C58PBX 71720415 IC50 = 7.5 nM T02562 C7TO8Z 71720734 IC50 = 910 nM T02562 C21ARQ 71720735 IC50 = 200 nM T02562 C04HXO 71748098 IC50 = 8.5 nM T02562 C8HZ6U 71764503 IC50 > 10000 nM T02562 CNY6H5 71765923 IC50 = 9.09 nM T02562 C71YGS 71765924 IC50 = 13.4 nM T02562 CYF2O1 71765925 IC50 = 11.3 nM T02562 CA4GY5 71766069 IC50 = 18.53 nM T02562 C7NKG8 71766070 IC50 = 249.9 nM T02562 CLZV93 71766071 IC50 = 14.34 nM T02562 CS46LC 71766073 IC50 = 7.2 nM T02562 C4AF1N 71766213 IC50 = 26.69 nM T02562 CB6J5U 71766365 IC50 = 15.25 nM T02562 CE3UF1 71766367 IC50 = 27.82 nM T02562 C1U7KS 71766510 IC50 = 18.66 nM T02562 CXAT19 71766651 IC50 = 49.47 nM T02562 CEU70M 71766652 IC50 = 64.3 nM T02562 CABU92 71766653 IC50 = 70.96 nM T02562 CDK1Y6 71766654 IC50 = 103.3 nM T02562 C51CDE 71766792 IC50 = 70.85 nM T02562 C7RV9H 71766793 IC50 = 4.19 nM T02562 C9PY8L 71766794 IC50 = 71.82 nM T02562 C5I8AY 71766795 IC50 = 141.2 nM T02562 CY9VC2 71766796 IC50 = 43.1 nM T02562 CKL41J 71766940 IC50 = 415.1 nM T02562 CUB64C 72546190 IC50 = 640 nM T02562 COI3K8 72548264 IC50 > 50000 nM T02562 CPB90G 72548265 IC50 = 7300 nM T02562 CMFD46 72734874 IC50 = 700 nM T02562 C2K0GM 72734875 IC50 = 1200 nM T02562 CBO3D4 72734876 IC50 = 1400 nM T02562 CUH2V3 72734877 IC50 = 1400 nM T02562 CD82PY 72734878 IC50 = 2300 nM T02562 CZWL24 72734879 IC50 = 500 nM T02562 C6WKI3 72735052 IC50 = 800 nM T02562 C3QIV9 72735053 IC50 = 700 nM T02562 CXZ2Q1 72735054 IC50 = 800 nM T02562 CPN87X 72735055 IC50 = 1700 nM T02562 C4TLU8 72735056 IC50 = 400 nM T02562 CWHB65 72735057 IC50 = 1600 nM T02562 CZB62X 72735237 IC50 = 1800 nM T02562 CU07KO 72735238 IC50 = 5000 nM T02562 CKH6N5 72735239 IC50 = 400 nM T02562 CQBP32 72735240 IC50 = 300 nM T02562 C9OXI7 72735241 IC50 = 400 nM T02562 C1DI9G 72735242 IC50 = 400 nM T02562 CWU6C4 72735414 IC50 = 500 nM T02562 CFNK27 72735415 IC50 = 1300 nM T02562 CB3SU5 72735416 IC50 = 900 nM T02562 CF8N6W 72735417 IC50 = 700 nM T02562 CX2ND4 72735418 IC50 = 1300 nM T02562 CVX16U 72735589 IC50 = 1700 nM T02562 CSDF35 72735590 IC50 = 600 nM T02562 C4JSP6 72735591 IC50 = 1900 nM T02562 CH5CF9 72735592 IC50 = 600 nM T02562 CG9JU0 72735593 IC50 = 600 nM T02562 C1XO0B 72735972 IC50 = 7200 nM T02562 CSOL63 72735973 IC50 = 1700 nM T02562 C7E1GS 72735974 IC50 = 1000 nM T02562 C5IYF9 72736361 IC50 = 800 nM T02562 CWJS67 72793857 IC50 = 80 nM T02562 CPDL08 73052732 IC50 = 300 nM T02562 C2RZ8J 73052890 IC50 = 180 nM T02562 CTY72V 73052891 IC50 = 680 nM T02562 CKR84E 73052892 IC50 = 810 nM T02562 CKC43H 73052893 IC50 = 430 nM T02562 C2B4OF 73053041 IC50 = 650 nM T02562 C16YKH 73053042 IC50 = 480 nM T02562 C7INR4 73356550 IC50 = 1500 nM T02562 CEM2R9 76324599 IC50 = 4000 nM T02562 CEO27D 86664693 IC50 = 9.6 nM T02562 C1EQP7 86664694 IC50 = 3.1 nM T02562 C9BCK4 86664703 IC50 = 4.7 nM T02562 C3HDU7 87424685 IC50 = 12 nM T02562 CSE81W 87570856 IC50 = 49 nM T02562 C9L2TE 88921783 IC50 = 7.76 nM T02562 C8MV7O 88921814 IC50 = 31.5 nM T02562 CH2JX8 88921834 IC50 = 21.02 nM T02562 CDM8H7 89854749 IC50 = 77.55 nM T02562 C3MZL7 89863688 IC50 = 12.53 nM T02562 CD1L4M 90643930 IC50 > 50000 nM T02562 C1Z7VS 90643931 IC50 > 50000 nM T02562 C9A6DF 90643932 IC50 > 50000 nM T02562 C84YLF 90643933 IC50 = 150 nM T02562 CD38OH 90643934 IC50 > 50000 nM T02562 C2TXO6 90643935 IC50 > 50000 nM T02562 CYLW90 90644054 IC50 = 4160 nM T02562 CKO9W2 90644055 IC50 = 7560 nM T02562 CS18JQ 90644056 IC50 > 30000 nM T02562 CSI21P 90644329 IC50 > 10000 nM T02562 C7N8YE 90644330 IC50 = 8500 nM T02562 C0Q2XP 90644331 IC50 = 10000 nM T02562 CDX79W 90644332 IC50 = 900 nM T02562 C07VSO 90644333 IC50 = 400 nM T02562 CEF51J 90644334 IC50 = 1200 nM T02562 CBXH26 90644335 IC50 = 400 nM T02562 C9EO0N 90644336 IC50 > 10000 nM T02562 CQG56R 90644337 IC50 = 1000 nM T02562 CR16AP 101909177 IC50 = 700 nM T02562 C82IOB 102161999 IC50 = 2800 nM T02562 CIRM37 118708871 IC50 > 10000 nM T02562 C7KJO8 118726052 IC50 = 5600 nM T02562 C3S9HT 118726053 IC50 = 1400 nM T02562 C2Z0RB 118726054 IC50 = 410 nM T02562 C6XH0K 118726938 IC50 = 5600 nM T02562 CE7L6H 118726939 IC50 = 5000 nM T02562 CB23OM 118726943 IC50 = 4900 nM T02562 CVU2B8 118726944 IC50 = 1600 nM T02562 C7EU9N 118726945 IC50 > 10000 nM T02562 CMS2J7 118726947 IC50 = 9200 nM T02562 CHM38G 118726948 IC50 > 10000 nM T02562 CY3J0G 118726949 IC50 = 3000 nM T02562 CR6IC4 118726951 IC50 = 10000 nM T02562 C4J5EW 118726952 IC50 = 8700 nM T02562 CVO6Y5 118726954 IC50 > 10000 nM T02562 CA8TS2 118726955 IC50 = 2500 nM T02562 C89LIX 118726956 IC50 = 3100 nM T02562 C18QZD 118726957 IC50 = 2400 nM T02562 CHA3C9 118987004 IC50 < 3 nM T02562 CD4Z7C 121313704 IC50 = 2 nM T02562 C1S5IC 121313869 IC50 = 7 nM T02562 CWL65U 121313879 IC50 = 12 nM T02562 C96YUN 121313880 IC50 = 1 nM T02562 CMW20L 121313882 IC50 = 30 nM T02562 CIKF48 121313888 IC50 = 3 nM T02562 CQV1W2 121313890 IC50 = 3 nM T02562 C7D6IX 121416984 IC50 = 10 nM T02562 C3NRT0 121416986 IC50 = 20 nM T02562 CB23CY 121417020 IC50 = 18 nM T02562 CTIG71 121417054 IC50 = 46 nM T02562 CV3W5D 121417061 IC50 = 30 nM T02562 C28OHG 121417086 IC50 = 32 nM T02562 CA53MF 121417157 IC50 = 15 nM T02562 CAC10H 121417161 IC50 = 569 nM T02562 CL05VT 121417168 IC50 = 22 nM T02562 CO78KD 121417175 IC50 = 30 nM T02562 C65DXP 121417176 IC50 = 961 nM T02562 CRH9G7 121417199 IC50 = 69 nM T02562 CA1Z2C 121417226 IC50 = 35 nM T02562 CRE8H4 121417251 IC50 = 208 nM T02562 CTSW21 121417260 IC50 = 161 nM T02562 CWP7Y2 121417263 IC50 = 29 nM T02562 CQ36IS 121417264 IC50 = 14 nM T02562 CE9XJ2 121426852 IC50 = 245 nM T02562 CP8GQ2 121426856 IC50 = 60 nM T02562 CV20KU 121426879 IC50 = 162 nM T02562 C96OQK 121426899 IC50 = 579 nM T02562 C1ZB0W 121426906 IC50 = 299 nM T02562 CIR0F1 121426923 IC50 = 72 nM T02562 C3R1VP 121426960 IC50 = 46 nM T02562 C4QW2G 121426971 IC50 = 70 nM T02562 CG2UF6 122185529 IC50 = 1 nM T02562 C0GFO5 122185605 IC50 = 500 nM T02562 CR2A4G 122185606 IC50 > 10000 nM T02562 C64DUW 122186832 IC50 = 5000 nM T02562 CTD1Q4 122186833 IC50 = 240 nM T02562 C0RTQ5 122186834 IC50 = 290 nM T02562 C9W7SY 122186835 IC50 = 220 nM T02562 CQBF95 122186836 IC50 = 390 nM T02562 C7U5XI 122186837 IC50 = 6400 nM T02562 CMGL28 122186838 IC50 = 610 nM T02562 C8Z5MV 122186839 IC50 = 680 nM T02562 CXT1Y6 122186841 IC50 = 570 nM T02562 C7C0JB 122186842 IC50 = 3500 nM T02562 CBH2L6 122186843 IC50 = 810 nM T02562 CIT2U6 122191352 IC50 > 30000 nM T02562 CE8P5N 122191353 IC50 > 30000 nM T02562 CH8IX0 122191354 IC50 > 30000 nM T02562 C6SCL2 122191355 IC50 > 30000 nM T02562 CDN0A3 123278303 IC50 = 92.94 nM T02562 CLTG52 124219472 IC50 = 43 nM T02562 C58KFT 124219480 IC50 = 1 nM T02562 CTG8S1 127025226 IC50 = 19.5 nM T02562 CJF07E 127025527 IC50 < 3 nM T02562 C71TBA 127026107 IC50 = 2000 nM T02562 CF4O7N 127026108 IC50 = 2000 nM T02562 CA6Z0B 127026109 IC50 = 2000 nM T02562 CI72YM 127026110 IC50 = 2000 nM T02562 C2CV9A 127027383 IC50 = 1330 nM T02562 CXLR24 127027708 IC50 = 13840 nM T02562 C84IUE 127027711 IC50 = 1930 nM T02562 C2RQC3 127028447 IC50 = 6.918 nM T02562 CY0VN8 127028780 IC50 = 5.012 nM T02562 C1P9GO 127028781 IC50 = 3.981 nM T02562 CEZL27 127029281 IC50 = 2000 nM T02562 CPBD98 127029537 IC50 = 2000 nM T02562 CNP78W 127029538 IC50 = 1020 nM T02562 C40GCD 127029539 IC50 = 2000 nM T02562 CS05BQ 127037918 IC50 > 10000 nM T02562 COQ8H2 127037919 IC50 > 10000 nM T02562 CB2TJ6 127038621 IC50 > 10000 nM T02562 CIS68G 127038622 IC50 > 10000 nM T02562 CI01ZD 127038623 IC50 = 6600 nM T02562 C12SUP 127038624 IC50 > 10000 nM T02562 CMZ7J4 127038975 IC50 = 70 nM T02562 CL0DU1 127038977 IC50 > 10000 nM T02562 CUC79J 127042501 IC50 = 6100 nM T02562 C4OI5E 127042537 IC50 > 10000 nM T02562 CU8LR4 132055261 IC50 = 3 nM T02562 C68WCR 132055288 IC50 = 1 nM T02562 C8ZH4A 132055290 IC50 = 2 nM T02562 CM83HC 132055304 IC50 = 1 nM T02562 C0DFT9 132055321 IC50 = 6 nM T02562 CLO7B9 132055329 IC50 = 2 nM T02562 CB9RO2 132055338 IC50 = 1 nM T02562 CYJP35 132055344 IC50 = 6 nM T02562 C1VN5Z 132079847 IC50 = 8 nM T02562 CA9JM4 132223627 IC50 = 44 nM T02562 CZ9SV2 132223628 IC50 = 15 nM T02562 C5N3GH 132223635 IC50 = 69 nM T02562 CQ1RE6 132223657 IC50 = 381 nM T02562 CUR9B4 134129928 IC50 = 9700 nM T02562 C0C2MB 134132426 IC50 = 46.6 nM T02562 CXFK72 134139665 IC50 = 4500 nM T02562 C1O5PR 134139870 IC50 = 10.79 nM T02562 C2XGP0 134141201 IC50 = 6 nM T02562 C9LH2U 134141703 IC50 = 15840 nM T02562 CYO40M 134146838 IC50 = 3720 nM T02562 CBUX92 134146911 IC50 = 14.65 nM T02562 C4HN2Y 134155900 IC50 = 6300 nM T02562 CYCO90 135419964 IC50 = 1800 nM T02562 C9IM4Z 135572096 IC50 = 5000 nM T02562 CPLD67 135798125 IC50 = 1 nM T02562 C3N2FJ 135906278 IC50 = 4500 nM T02562 CR67MD 136042253 IC50 = 4116 nM T02562 CG16FT 136044208 IC50 = 36 nM T02562 CN2I5U 136044209 IC50 = 26 nM T02562 C67WKO 136044210 IC50 = 63 nM T02562 C5V3JS 136044211 IC50 = 7 nM T02562 CD5U1M 136044212 IC50 = 74 nM T02562 CP0Y9W 136044213 IC50 = 36 nM T02562 C6V5JM 136044214 IC50 = 32 nM T02562 CW4C9D 136044215 IC50 = 111 nM T02562 C2IYU6 136044216 IC50 = 261 nM T02562 CJQT13 136044217 IC50 = 24 nM T02562 CBMU49 136044218 IC50 = 481 nM T02562 CQS60T 136044219 IC50 = 243 nM T02562 CI63QS 136056624 IC50 > 50000 nM T02562 CSK95Y 136504263 IC50 = 13 nM T02562 C0Y4AH 137632562 IC50 = 461 nM T02562 CPNL17 137632852 IC50 = 2 nM T02562 C2HES1 137634058 IC50 = 1200 nM T02562 CFV73H 137637242 IC50 = 276 nM T02562 C72SBZ 137638298 IC50 = 56.89 nM T02562 CKL6R0 137638693 IC50 = 664 nM T02562 CI6N9P 137642063 IC50 = 1000 nM T02562 CUH75A 137648374 IC50 = 73.89 nM T02562 C7QKU0 137649316 IC50 = 439 nM T02562 C3F7GH 137649890 IC50 = 5340 nM T02562 CTCY45 137649934 IC50 = 1100 nM T02562 C3MDL6 137652327 IC50 = 284 nM T02562 CHI80F 137652936 IC50 > 10000 nM T02562 C92CGQ 137655546 IC50 = 2400 nM T02562 CA39BM 137655857 IC50 = 889 nM T02562 C8CZ1B 137659631 IC50 = 2400 nM T02562 CBK0G4 137660563 IC50 = 187.3 nM T02562 CQE5X9 145432862 IC50 = 622 nM T02562 C0KT9F 145432921 IC50 = 285 nM T02562 C3Q7HY 145432944 IC50 = 169 nM T02562 C34MVG 145432945 IC50 = 212 nM T02562 CM7AN9 145432972 IC50 = 265 nM T02562 CLR3Z7 145949593 IC50 = 2800 nM T02562 C65VCJ 145959226 IC50 = 2000 nM T02562 C3KFX8 145963880 IC50 = 36 nM T02562 CIT37R 145964590 IC50 = 1590 nM T02562 CLXW39 145964963 IC50 = 7.7 nM T02562 CHNP84 145965699 IC50 = 92 nM T02562 CWY1L2 145966759 IC50 = 83 nM T02562 C9K4CF 145967020 IC50 = 4.2 nM T02562 C0P3IA 145967142 IC50 = 361 nM T02562 C6CV8W 145968005 IC50 = 561 nM T02562 C5I1JL 145968680 IC50 = 20 nM T02562 CU56JO 145970054 IC50 = 337 nM T02562 CE5B8S 145971409 IC50 = 1040 nM T02562 CB5EA8 145971903 IC50 = 1390 nM T02562 CU1L0J 145972089 IC50 = 52 nM T02562 CP0F4E 145974651 IC50 = 294 nM T02562 CBX70R 145975131 IC50 = 95 nM T02562 CZA0V2 145975174 IC50 = 56 nM T02562 C3B9RX 145975918 IC50 = 598 nM T02562 C3UZ2T 145975940 IC50 = 797 nM T02562 CBQ58M 145977002 IC50 = 283 nM T02562 CE5N9D 145977523 IC50 = 93 nM T02562 C81EIF 145978189 IC50 = 41 nM T02562 CA2HL1 145978765 IC50 = 1730 nM T02562 C7OJS3 145978845 IC50 = 92 nM T02562 CO8RY0 145978927 IC50 = 1100 nM T02562 C2NUH7 145979828 IC50 = 700 nM T02562 C7G6DE 145980236 IC50 = 600 nM T02562 COYB38 145980268 IC50 = 58800 nM T02562 CLCU07 145980449 IC50 = 180 nM T02562 CMRJ31 145980727 IC50 = 5300 nM T02562 CXN01G 145980737 IC50 = 1640 nM T02562 CM73GH 145981036 IC50 = 6200 nM T02562 CO84KR 145981339 IC50 = 2130 nM T02562 CM02LY 145981376 IC50 = 5000 nM T02562 C3EDP1 145982139 IC50 = 5400 nM T02562 C4OPU2 145982203 IC50 > 10000 nM T02562 CZQY07 145982329 IC50 = 6500 nM T02562 CH3GA6 145982419 IC50 = 2560 nM T02562 C1IBC7 145983185 IC50 = 3200 nM T02562 CU95NM 145983649 IC50 = 420 nM T02562 CF82BO 145984396 IC50 > 10000 nM T02562 CM62SF 145985303 IC50 = 2100 nM T02562 CQ0F4H 145986097 IC50 = 1200 nM T02562 CH1TE6 145986374 IC50 = 4700 nM T02562 C85VGU 145986619 IC50 > 10000 nM T02562 C5VJ0U 145986782 IC50 = 4700 nM T02562 CT7NK0 145986883 IC50 = 260 nM T02562 C5V4BG 145986923 IC50 = 4200 nM T02562 CVA7K0 145986989 IC50 = 3430 nM T02562 C4ZBC9 145987188 IC50 = 1900 nM T02562 CG2J7C 145987315 IC50 = 5200 nM T02562 C20LTV 145987586 IC50 = 1190 nM T02562 CU03MH 145987714 IC50 = 3800 nM T02562 CYX25Q 145987750 IC50 > 10000 nM T02562 C7DWP8 145988191 IC50 = 7060 nM T02562 CE15SN 145988338 IC50 = 12700 nM T02562 C10NDO 145988652 IC50 = 2540 nM T02562 C8SVA1 145989549 IC50 = 4000 nM T02562 C1SF0G 145989884 IC50 = 540 nM T02562 CU1ET5 145990280 IC50 = 1000 nM T02562 CM8K2G 145990428 IC50 = 4200 nM T02562 C0YFW7 145991004 IC50 = 2700 nM T02562 CRJ35U 145991263 IC50 > 10000 nM T02562 CA69OZ 145991533 IC50 = 3400 nM T02562 CJ23ZQ 145991963 IC50 = 8600 nM T02562 C14RPI 145992031 IC50 = 300 nM T02562 CQ39BP 145992502 IC50 = 2900 nM T02562 C38CIQ 145992873 IC50 = 480 nM T02562 C7QZ9D 145993245 IC50 = 1600 nM T02562 CQL0D9 145993288 IC50 = 2700 nM T02562 CN8G1X 145993375 IC50 = 700 nM T02562 CU80CE 145993587 IC50 = 1900 nM T02562 CNUM28 145994201 IC50 = 6300 nM T02562 C67STF 155510868 IC50 = 9260 nM T02562 CXJT08 155511272 IC50 = 21 nM T02562 CA2Z5R 155514695 IC50 = 9740 nM T02562 CNS2M6 155516585 IC50 = 11300 nM T02562 CWC54X 155521712 IC50 = 327 nM T02562 CS6LY3 155523181 IC50 = 2330 nM T02562 CA3VU5 155525210 IC50 > 20000 nM T02562 CPV37A 155525752 IC50 = 270 nM T02562 C1G0CE 155525854 IC50 = 980 nM T02562 C67DJL 155527581 IC50 = 10 nM T02562 CL23MT 155529344 IC50 = 276 nM T02562 C7HD4B 155529702 IC50 > 20000 nM T02562 CHY87X 155530077 IC50 > 20000 nM T02562 CBP3S1 155532334 IC50 > 20000 nM T02562 CE0J1G 155532421 IC50 = 1960 nM T02562 CNZ70R 155533624 IC50 = 7030 nM T02562 CUZ2T5 155536736 IC50 = 670 nM T02562 C92RYO 155536880 IC50 > 20000 nM T02562 CNHC78 155544254 IC50 > 20000 nM T02562 C0BMX4 155545361 IC50 = 371 nM T02562 C9FP7Q 155546635 IC50 = 5860 nM T02562 C6KBO3 155547839 IC50 = 3090 nM T02562 CV8EP4 155549875 IC50 = 752 nM T02562 C5LMN1 155550498 IC50 = 8510 nM T02562 C1ZR7L 155551578 IC50 = 4490 nM T02562 CPQW25 155552628 IC50 = 10600 nM T02562 CR7I9W 155557497 IC50 > 20000 nM T02562 CJC27Y 155560410 IC50 > 20000 nM T02562 CBUJ49 155569147 IC50 = 152 nM T02562 D02XEX 11168203 IC50 = 3000 nM T02562 D06TXM 24816385 IC50 = 3400 nM T02562 D09VTJ 441298 IC50 = 1000 nM T02562 D09VYW 9847548 IC50 = 3000 nM T02562 D0IR6U 5494425 IC50 > 10000 nM T02562 D0W6TB 16730275 IC50 = 1 nM T84981 D0YQ7U 11285792 IC50 = 3.1 nM T84981 D0W0LS 183789 IC50 = 1.4 nM T84981 C06TUD 11285791 IC50 > 10000 nM T84981 C8E3GU 26042546 IC50 > 30000 nM T84981 C6ENV5 100951623 EC50 > 10000 nM T84981 C5I8EN 134817249 IC50 = 9400 nM T84981 C4Z3XS 145983516 IC50 > 30000 nM T84981 C9NDM5 145983631 IC50 > 30000 nM T84981 C3ZPR5 145985518 IC50 > 30000 nM T84981 CHTY23 145985766 IC50 = 18000 nM T84981 D06MBD 11176403 IC50 > 3000 nM T22939 D04DJN 10635 EC50 = 8200 nM T22939 D07BSQ 5994 EC50 = 0.1 nM T22939 D07KSG 2733526 IC50 = 128.82 nM T22939 D0BC2E 91649 IC50 = 2013 nM T22939 D0D1SG 5755 Ki > 1000 nM T22939 D0EP0C 5833 Ki = 399.7 nM T22939 D0F2AK 36709 IC50 = 0.236 nM T22939 D0G8BV 6450278 Ki = 224 nM T22939 D0GL7U 6230 Ki = 1.87 nM T22939 D0IT2G 5743 IC50 = 440 nM T22939 D0JO7Y 104741 IC50 = 0.2089 nM T22939 D0Q4SD 443872 IC50 > 10000 nM T22939 D0V9BD 2375 IC50 = 1819 nM T22939 D0Y7IU 5281004 IC50 = 28 nM T22939 D0Y7JU 9854489 IC50 = 21 nM T22939 D0Z4EI 55245 IC50 = 0.025 nM T22939 D00JFE 56941241 IC50 > 1000 nM T22939 D01SYU 10026128 IC50 = 10000 nM T22939 D07MON 5311505 EC50 = 1.6 nM T22939 D09ZLZ 44200882 IC50 = 750 nM T22939 D0HE7C 134415769 IC50 = 21 nM T22939 D0L3HU 6918548 IC50 = 0.0025 nM T22939 D0SZ1G 121248172 IC50 = 5300 nM T22939 D0X1OW 86287635 IC50 = 540 nM T22939 D0X9YP 67041274 IC50 > 10000 nM T22939 D0TH6M 25204767 EC50 > 10000 nM T22939 D02KAU 46871935 IC50 = 416 nM T22939 D03KTE 16750192 Ki = 2500 nM T22939 D09UFV 24825740 IC50 = 1760 nM T22939 D0L5KF 132981 IC50 = 1000 nM T22939 D0W5RL 9577221 IC50 = 0.3 nM T22939 C59UQE 6279 EC50 = 0.1 nM T22939 C0XDJ1 9880 IC50 > 1000 nM T22939 CQ0IC4 63062 IC50 = 0.7943 nM T22939 CB14QJ 130904 IC50 = 0.2 nM T22939 CJA6Z2 242636 IC50 = 84000 nM T22939 C40YBS 444036 IC50 = 21 nM T22939 CKZN26 603699 IC50 = 1700 nM T22939 C2B0JA 674359 Ki = 147 nM T22939 C4GKV7 744859 IC50 = 2800 nM T22939 C0U4FD 786364 IC50 = 2200 nM T22939 CB02WA 889300 IC50 = 1300 nM T22939 CQ93FY 889795 IC50 = 820 nM T22939 CGIL56 1484235 IC50 > 1000 nM T22939 C6YHO1 1484236 IC50 = 416 nM T22939 CEJ9K4 1484237 IC50 = 521 nM T22939 CGD23L 1834356 EC50 = 199.53 nM T22939 CP3RV7 1834359 IC50 = 6309.57 nM T22939 C57UHE 2255761 IC50 = 8100 nM T22939 CJ6FL4 2325104 IC50 = 4900 nM T22939 C3BM0D 2348480 IC50 = 520 nM T22939 C0YO8A 2876244 IC50 = 140 nM T22939 CTBC06 2941086 EC50 = 630.96 nM T22939 CQXE70 2952744 IC50 = 1258.93 nM T22939 C2EHS5 2952945 IC50 = 794.33 nM T22939 C0CUX1 3160911 EC50 > 10000 nM T22939 C6YZV8 3160913 EC50 > 10000 nM T22939 CCH1G5 3160915 EC50 = 3981.07 nM T22939 CNC1R7 3160916 EC50 > 10000 nM T22939 CHSE72 3272891 IC50 = 500 nM T22939 C47TUA 3330197 IC50 = 17000 nM T22939 CLBV35 3699263 IC50 > 2000 nM T22939 C56BXH 3775890 IC50 = 84 nM T22939 C43BVE 3816305 IC50 > 2000 nM T22939 CUP17G 3831396 IC50 = 62.4 nM T22939 CF1E6B 3865807 IC50 = 1500 nM T22939 CZA46J 4111936 IC50 = 1300 nM T22939 C9Q2VK 4180255 IC50 = 26000 nM T22939 CL0P5X 5067753 IC50 = 10000 nM T22939 CB1CK8 5157385 IC50 = 670 nM T22939 CDCK27 5185174 IC50 = 1000 nM T22939 CJB7T6 5288494 IC50 = 3981.07 nM T22939 C16ZSG 6439929 Ki = 201 nM T22939 CNLU79 8029772 IC50 = 34000 nM T22939 CKA32J 8190105 IC50 = 1300 nM T22939 CK6LQ1 8512912 IC50 = 1600 nM T22939 CI9Q8R 9795365 IC50 = 102 nM T22939 C1Q2TS 9795451 IC50 = 3.8 nM T22939 CO46RD 9795931 IC50 = 642 nM T22939 CRW95K 9796472 EC50 = 1.7 nM T22939 C3V0OT 9802328 Ki = 0.59 nM T22939 C7REX1 9805004 IC50 = 19 nM T22939 C5GY8B 9814216 IC50 = 8 nM T22939 CFGH58 9814351 IC50 = 19.5 nM T22939 C5US4R 9816921 IC50 = 66 nM T22939 CT73GV 9817870 IC50 = 6.6 nM T22939 CTD7Q2 9818809 EC50 = 1.6 nM T22939 CV87EA 9820084 IC50 = 1400 nM T22939 C8A3WG 9820510 Ki = 7000 nM T22939 C06RXB 9821393 Ki > 5000 nM T22939 C7HGB0 9822150 Ki = 0.55 nM T22939 CD9S5P 9825465 Ki > 5000 nM T22939 CT6OZ1 9825650 IC50 > 1000 nM T22939 C6B3ST 9836954 EC50 = 1 nM T22939 CIXV16 9837713 IC50 = 296 nM T22939 CM9C2V 9838980 EC50 = 60 nM T22939 CE62WD 9839013 Ki = 10 nM T22939 CGZW90 9839078 EC50 = 0.4 nM T22939 CBS8M2 9839134 IC50 = 15.9 nM T22939 CO5M2U 9839495 EC50 = 500 nM T22939 C92CPK 9841404 Ki = 5300 nM T22939 CK7UC3 9841413 Ki = 5400 nM T22939 C7P6XH 9842832 Ki = 2800 nM T22939 CE9A6G 9845022 Ki = 0.49 nM T22939 C7RS9U 9846657 Ki = 1560 nM T22939 CZ2E1D 9851926 IC50 = 10 nM T22939 C0TQW2 9860141 IC50 = 300 nM T22939 C2Y5NU 9860277 IC50 = 130 nM T22939 C7M1IG 9860721 IC50 = 300 nM T22939 CWI42R 9860776 IC50 = 29 nM T22939 CERF28 9861044 Ki = 5200 nM T22939 C3K4EU 9862027 Ki > 10000 nM T22939 CH5GT6 9862037 Ki = 1.9 nM T22939 CJN78I 9862597 EC50 = 0.36 nM T22939 C98JAL 9878929 EC50 ~ 1000 nM T22939 CWX20S 9878992 IC50 = 180 nM T22939 CWV2Y4 9879853 IC50 = 26.2 nM T22939 CX4K8J 9882391 IC50 = 9.3 nM T22939 C01ZFV 9882789 IC50 > 10000 nM T22939 C6R5XE 9884128 IC50 = 412 nM T22939 CEM27C 9885473 Ki = 4.9 nM T22939 C8XSO2 9887578 Ki = 0.1 nM T22939 C6B9CZ 9888873 IC50 = 30 nM T22939 CZ5R9B 9890023 Ki = 4000 nM T22939 CCM30W 9901180 Ki > 5000 nM T22939 CNH12G 9903346 Ki = 127 nM T22939 C6X4LN 9903502 IC50 = 1529 nM T22939 COC71W 9903853 EC50 = 1.1 nM T22939 CN3T2F 9904225 EC50 = 1.8 nM T22939 CJ7U3R 9904286 IC50 = 200 nM T22939 CWK42S 9904407 IC50 = 27 nM T22939 C4KY8S 9904429 EC50 = 0.38 nM T22939 C6SWK1 9904610 IC50 = 23 nM T22939 C65ZOT 9904865 EC50 = 0.6 nM T22939 CY2Q4D 9905086 EC50 = 2 nM T22939 CTI1J8 9905296 Ki = 2000 nM T22939 CN9R3V 9906170 IC50 = 62 nM T22939 CE1TK2 9908041 Ki = 0.83 nM T22939 CVN0H9 9909625 EC50 = 2.8 nM T22939 CMJG42 9921530 IC50 = 40.2 nM T22939 C49UGC 9925244 Ki = 1700 nM T22939 CBGV39 9925534 Ki = 19 nM T22939 C4CJ6A 9925757 IC50 = 30.6 nM T22939 CBZ15C 9926184 IC50 = 15 nM T22939 C8MKC4 9926926 EC50 = 200 nM T22939 C39EXP 9933936 IC50 = 10000 nM T22939 C24FUO 9943699 IC50 = 6.7 nM T22939 CXM67A 9946466 Ki > 5000 nM T22939 CAR6G1 9947862 EC50 = 5 nM T22939 C5C6HA 9947878 IC50 = 20.6 nM T22939 CZVR83 9948117 IC50 = 330 nM T22939 C3X7CJ 9948246 IC50 = 229 nM T22939 C5QF9L 9948250 EC50 = 28.7 nM T22939 CST95Z 9949175 EC50 = 0.3 nM T22939 CCSX75 9949772 IC50 = 210 nM T22939 C6ZT3M 9950357 IC50 = 460 nM T22939 CKU64T 9952569 IC50 = 236 nM T22939 CW0ED9 9953456 EC50 = 2.1 nM T22939 CN50BQ 9964788 IC50 ~ 3000 nM T22939 C4GP8K 9965224 EC50 ~ 3000 nM T22939 CEM8L7 9969737 Ki > 5000 nM T22939 C0Y1RE 9969849 Ki = 610 nM T22939 CBLF36 9973351 IC50 = 5.7 nM T22939 C95CAN 9978625 Ki = 15.5 nM T22939 CP2E8A 9979395 EC50 = 35 nM T22939 C1QP8T 9993897 IC50 = 1900 nM T22939 C7R0QI 9994029 EC50 = 1.25 nM T22939 CGH6Z0 9994920 EC50 = 7.2 nM T22939 C03NHV 9995323 Ki = 3.6 nM T22939 CXC8K1 9995611 EC50 = 1.6 nM T22939 CWRV14 9996069 EC50 = 42 nM T22939 COA3P9 9997031 IC50 > 2000 nM T22939 C47RUV 9998207 IC50 = 620 nM T22939 C4V6RF 9998996 IC50 > 1000 nM T22939 CU1ON0 9999068 Ki = 7.6 nM T22939 CL8V1C 9999671 IC50 = 1600 nM T22939 CU4L7C 9999672 IC50 > 2000 nM T22939 C08OBS 10001663 IC50 > 2000 nM T22939 C0XDE9 10001914 IC50 > 2000 nM T22939 C69CGV 10016740 Ki = 28 nM T22939 CE7L5G 10017966 EC50 = 1.5 nM T22939 C3G0SD 10020808 IC50 = 17 nM T22939 C3IE9K 10021634 IC50 = 330 nM T22939 CKC56N 10021648 EC50 = 1200 nM T22939 CJ0O2X 10021826 IC50 > 2000 nM T22939 C52ADB 10023861 Ki = 3.5 nM T22939 CN8BH3 10024007 IC50 = 14 nM T22939 CC4WY6 10024990 IC50 = 440 nM T22939 CSM0W3 10026120 IC50 > 2000 nM T22939 C3GO1K 10040475 EC50 = 0.7 nM T22939 CWKY34 10042477 EC50 = 1.4 nM T22939 C3ITG8 10044396 IC50 > 2000 nM T22939 C9PE6Q 10045301 EC50 = 88.5 nM T22939 CK50XF 10048063 IC50 = 1200 nM T22939 CV7L3C 10064703 EC50 = 79.5 nM T22939 COM8R7 10065049 EC50 = 5.3 nM T22939 CE36CK 10065209 EC50 = 1000 nM T22939 C0MG6I 10067556 IC50 > 2000 nM T22939 C2V9BW 10068183 IC50 = 950 nM T22939 CJ9K8H 10068202 IC50 = 100 nM T22939 CJ0C5D 10070462 IC50 = 0.073 nM T22939 CB5OZ0 10070722 IC50 > 2000 nM T22939 CFY67M 10070808 Ki = 2.6 nM T22939 C7JQM6 10070842 IC50 > 2000 nM T22939 C9T4HR 10071810 IC50 > 2000 nM T22939 C5MR6U 10071910 IC50 = 1000 nM T22939 CLO7H6 10072320 IC50 = 1900 nM T22939 CNP1M6 10086357 EC50 = 49.8 nM T22939 C0J5BO 10086987 EC50 = 1.1 nM T22939 C8CDS0 10087446 EC50 = 0.9 nM T22939 CRG90H 10088261 EC50 = 2.5 nM T22939 CQ3LD1 10091351 IC50 = 170 nM T22939 C2C7NE 10091387 IC50 > 2000 nM T22939 CRP4A3 10091735 IC50 > 2000 nM T22939 C16HAK 10094808 IC50 > 2000 nM T22939 CVC7S6 10108111 EC50 = 11.6 nM T22939 CWR57A 10113229 Ki > 5000 nM T22939 C62CGR 10125859 Ki > 5000 nM T22939 CM4DK2 10125966 Ki = 760 nM T22939 CDBJ41 10126018 Ki > 5000 nM T22939 CO97CW 10126196 Ki > 5000 nM T22939 CR0DX5 10126475 IC50 > 1130 nM T22939 CHS18G 10126476 IC50 > 2000 nM T22939 CR0BP6 10126871 IC50 = 250 nM T22939 CV5PQ0 10126940 IC50 = 280 nM T22939 CVF40M 10127159 IC50 = 265 nM T22939 C3CRZ1 10127269 IC50 > 2000 nM T22939 CPB60D 10127340 IC50 > 2000 nM T22939 C1K8UF 10127593 IC50 = 30 nM T22939 C8VBQ0 10127709 IC50 = 40 nM T22939 CKMW98 10128037 IC50 = 415 nM T22939 C7CNX6 10128352 IC50 = 180 nM T22939 C1GI3D 10150743 IC50 > 354 nM T22939 CZKF71 10150825 IC50 = 225 nM T22939 CYR0U5 10150851 IC50 > 2000 nM T22939 CVO1F7 10151165 IC50 = 405 nM T22939 C6EC1P 10151186 IC50 = 710 nM T22939 CQ14RM 10151357 IC50 > 2000 nM T22939 C6U0FQ 10151473 IC50 = 47 nM T22939 CW4Y2K 10151995 IC50 = 1750 nM T22939 CDV0H3 10152035 IC50 = 48 nM T22939 CR6N7C 10156793 Ki = 349 nM T22939 C0MX7K 10157532 IC50 = 6896 nM T22939 CL0U4N 10172897 IC50 > 2000 nM T22939 C56RYS 10173217 IC50 = 240 nM T22939 CG0VH8 10173354 IC50 = 1800 nM T22939 CU6D8W 10173525 IC50 = 35 nM T22939 CP4Y6T 10173634 IC50 = 59 nM T22939 C14HMT 10173659 IC50 = 44 nM T22939 CE29WD 10174141 IC50 = 34 nM T22939 CU2IT3 10177239 Ki = 2.2 nM T22939 C8L7HJ 10179031 IC50 = 476 nM T22939 CHK2V6 10193599 Ki > 5000 nM T22939 C5SRU4 10193967 Ki > 5000 nM T22939 C41YRZ 10194268 IC50 > 740 nM T22939 CX4F7Z 10194607 IC50 > 2000 nM T22939 CV0LE4 10194889 IC50 = 1000 nM T22939 CJ1GX6 10195783 IC50 = 51 nM T22939 CRIH90 10210815 IC50 = 180 nM T22939 C8HDU9 10215137 Ki = 4300 nM T22939 C3O7WH 10215978 IC50 > 2000 nM T22939 CX6FD1 10216117 Ki > 5000 nM T22939 C1SG4N 10216152 IC50 > 1420 nM T22939 CD0YT7 10216465 IC50 > 2000 nM T22939 C1FGX9 10216535 IC50 = 350 nM T22939 CW7QX2 10216536 IC50 = 1250 nM T22939 CG9OH4 10216697 IC50 = 1200 nM T22939 CXN4W1 10216788 IC50 > 2000 nM T22939 CUGN98 10217411 IC50 = 1600 nM T22939 C3XK0O 10217420 IC50 = 36 nM T22939 C3TIU7 10220661 IC50 = 299 nM T22939 C6QO7E 10220791 IC50 = 1370 nM T22939 CJ2OG0 10220994 EC50 = 2.1 nM T22939 C54HJB 10221941 Ki > 5000 nM T22939 CJ9BE0 10222329 IC50 = 673 nM T22939 C84SRT 10223610 IC50 = 498 nM T22939 CUYO17 10237223 IC50 > 1600 nM T22939 C4KF2V 10237539 Ki > 5000 nM T22939 CWYK62 10238100 IC50 = 930 nM T22939 C1R8GY 10238297 IC50 = 1300 nM T22939 CNB1V3 10238624 IC50 = 35 nM T22939 CPGF94 10238831 IC50 > 2000 nM T22939 C2AZH1 10238961 IC50 = 330 nM T22939 C56PQZ 10247253 IC50 = 480 nM T22939 C7ZC3W 10248313 EC50 = 1.7 nM T22939 C7BMH6 10251407 IC50 = 7.1 nM T22939 CSA4R3 10252455 IC50 = 1400 nM T22939 C7EGH2 10252527 IC50 = 470 nM T22939 CR59SC 10271193 IC50 = 3355 nM T22939 CPIS57 10271557 IC50 = 450 nM T22939 CC4WT8 10272405 Ki = 1810 nM T22939 C9UL4O 10272529 Ki = 3740 nM T22939 CZP75A 10286964 Ki > 5000 nM T22939 CUQC81 10287415 IC50 > 1000 nM T22939 C5RC7X 10287444 IC50 = 345 nM T22939 CJT2G8 10287863 IC50 > 2000 nM T22939 C1M6WY 10288006 IC50 = 140 nM T22939 CO6UP3 10288155 IC50 = 665 nM T22939 CNT3V9 10288528 IC50 = 160 nM T22939 C6C2IK 10288565 IC50 = 80 nM T22939 C1I9JX 10288784 IC50 = 35 nM T22939 CNEO49 10289020 IC50 = 32 nM T22939 CLJU03 10298892 Ki > 5000 nM T22939 C9UYG8 10309447 IC50 > 1050 nM T22939 C8FM2D 10309755 IC50 > 2000 nM T22939 C1OV7M 10309756 IC50 > 2000 nM T22939 C9TI4A 10310063 IC50 = 1450 nM T22939 CP9AE0 10310476 IC50 > 512 nM T22939 CV52EN 10310809 IC50 = 42 nM T22939 CR1L5N 10311251 IC50 = 35 nM T22939 C9FCQ5 10313926 Ki = 4.467 nM T22939 CS3H6A 10314478 EC50 = 44.9 nM T22939 CUG85P 10314517 EC50 = 5.4 nM T22939 C7RLW3 10314903 IC50 > 2000 nM T22939 C4KYF1 10314964 EC50 = 14.8 nM T22939 C8HA2F 10315582 EC50 = 4.3 nM T22939 CX7WS4 10316069 Ki = 3.6 nM T22939 CR9ON2 10316670 IC50 = 1300 nM T22939 CZFY94 10318044 IC50 > 2000 nM T22939 CGVF38 10318898 IC50 = 100 nM T22939 CJB8R4 10319017 Ki = 1.3 nM T22939 C6J4AK 10319126 Ki = 0.32 nM T22939 C6OI7M 10336208 IC50 > 2000 nM T22939 CEB82Z 10337245 Ki = 34 nM T22939 C4QY5H 10337273 IC50 = 360 nM T22939 CS4J3T 10337784 EC50 = 2.5 nM T22939 C3PHW5 10339694 IC50 > 2000 nM T22939 C8IAJ7 10339824 IC50 > 2000 nM T22939 CK20PF 10339825 IC50 > 2000 nM T22939 CQP1Y7 10340204 Ki = 0.7 nM T22939 C28SWP 10341012 IC50 = 660 nM T22939 C9QUT6 10341919 IC50 = 210 nM T22939 CQ01DG 10342379 IC50 > 2000 nM T22939 CZ8N1T 10357739 EC50 = 1.5 nM T22939 CAV5E7 10359219 EC50 = 0.8 nM T22939 C61FVO 10360420 IC50 = 17.5 nM T22939 CEW79S 10361500 IC50 > 2000 nM T22939 CA20SQ 10362131 IC50 = 440 nM T22939 C2PSC1 10362449 IC50 > 2000 nM T22939 CMSA84 10362453 IC50 > 2000 nM T22939 CEJ78I 10365592 IC50 > 2000 nM T22939 C6QR5M 10366372 IC50 > 2000 nM T22939 CDBZ06 10372181 IC50 = 550 nM T22939 CH24CS 10379313 EC50 = 1 nM T22939 CA16IK 10380384 EC50 = 11.4 nM T22939 C40CJF 10380579 EC50 = 1.9 nM T22939 C2B3UC 10382522 EC50 = 0.5 nM T22939 C6HTP7 10383035 IC50 = 24 nM T22939 C64FYW 10383547 EC50 = 2.5 nM T22939 CKB19V 10383968 IC50 = 10 nM T22939 C14AIB 10384345 IC50 = 451 nM T22939 C6RQK1 10386584 IC50 > 10000 nM T22939 C2MIC7 10388043 IC50 = 1300 nM T22939 C25TXP 10403527 EC50 = 2.6 nM T22939 C3KRL5 10404759 EC50 = 1.4 nM T22939 CBU68V 10406413 Ki = 150 nM T22939 C3P1OZ 10406621 EC50 = 7.7 nM T22939 CEQW13 10407564 IC50 > 2000 nM T22939 CS5XF8 10408522 IC50 > 2000 nM T22939 C8ERB7 10411364 IC50 = 930 nM T22939 CZ5CJ3 10423330 Ki = 53.5 nM T22939 C2WHE6 10423425 EC50 = 300 nM T22939 CP5SL3 10424022 EC50 = 0.35 nM T22939 C01KVL 10426609 EC50 = 2000 nM T22939 CX5U9W 10427481 EC50 = 4.7 nM T22939 CQTX10 10427689 EC50 = 0.5 nM T22939 C3LF9D 10428026 IC50 > 2000 nM T22939 CJ6T4F 10428171 IC50 = 1600 nM T22939 CHR4W7 10429332 IC50 = 960 nM T22939 CL1E5U 10429892 EC50 = 23.5 nM T22939 C37VXR 10432143 IC50 = 354 nM T22939 C1KE6C 10446402 Ki = 3.467 nM T22939 C0VUS8 10446594 EC50 = 1.2 nM T22939 CHQ12T 10449284 EC50 = 0.3 nM T22939 CI91JZ 10450619 IC50 = 460 nM T22939 CU2WN9 10451276 IC50 = 100 nM T22939 CE31PF 10453033 EC50 = 80.1 nM T22939 C0NT9D 10454007 IC50 > 1000 nM T22939 C7OL9I 10455482 IC50 = 100 nM T22939 C1H5RP 10458842 EC50 > 10 nM T22939 CZ5P4J 10471922 EC50 = 7.2 nM T22939 CH8JI6 10472205 EC50 = 4.2 nM T22939 CHX67B 10472284 EC50 = 26.5 nM T22939 C28IGJ 10472499 EC50 = 2.6 nM T22939 CI46NV 10472986 EC50 = 5.7 nM T22939 C85RBN 10474264 IC50 = 1400 nM T22939 C1S9HE 10474749 IC50 = 980 nM T22939 CUL8O4 10475384 IC50 = 660 nM T22939 CN7KQ8 10475688 IC50 > 2000 nM T22939 C8O1QG 10476314 EC50 = 5.3 nM T22939 CPX65M 10477088 IC50 = 570 nM T22939 CDLT53 10494026 Ki = 19.95 nM T22939 CYE7C2 10496255 Ki = 71 nM T22939 C34YHX 10496434 IC50 = 1020 nM T22939 CT7IG5 10497270 Ki = 84 nM T22939 CZ2LN5 10499217 Ki = 2.1 nM T22939 CRC43Y 10499305 IC50 > 1000 nM T22939 CO35TR 10499308 IC50 = 2000 nM T22939 COH27F 10499475 Ki = 0.69 nM T22939 CCNU53 10500181 Ki = 5.6 nM T22939 CAZ30C 10501135 Ki = 1.3 nM T22939 CZU9R7 10501479 Ki = 0.34 nM T22939 C6FA1N 10501542 Ki = 98 nM T22939 C9A6YD 10502271 Ki = 10.8 nM T22939 CA5OH2 10503046 Ki = 0.5 nM T22939 C5AP6C 10503520 Ki = 0.87 nM T22939 C5WP1Q 10517398 IC50 = 94 nM T22939 C63ENM 10518992 IC50 = 231 nM T22939 CB0RC3 10520975 IC50 = 362 nM T22939 CI0ZD8 10522569 IC50 = 38.2 nM T22939 CR1OS9 10523126 EC50 = 9 nM T22939 CN5E6A 10523777 Ki = 39.7 nM T22939 C28FOD 10524140 Ki = 6.3 nM T22939 C5CDF0 10524606 IC50 = 210 nM T22939 C9H5IE 10525353 Ki = 2.7 nM T22939 CNW0F8 10525706 IC50 = 470 nM T22939 C2HG4R 10527530 Ki = 2.4 nM T22939 CKXU80 10542131 IC50 = 70.6 nM T22939 CYS8J9 10546095 IC50 = 1700 nM T22939 CI4ZX7 10546500 IC50 = 570 nM T22939 CP8A1M 10548404 EC50 = 48 nM T22939 CYB34C 10549156 Ki = 1.3 nM T22939 C9B2IH 10549288 IC50 = 460 nM T22939 CZ31QX 10567979 IC50 = 2200 nM T22939 C96GWO 10567980 IC50 = 1144 nM T22939 C87UQF 10568861 IC50 = 4395 nM T22939 C7G6IU 10570684 IC50 > 1000 nM T22939 CCOE17 10591908 IC50 = 233 nM T22939 CB04AE 10593144 Ki = 77 nM T22939 C5CZ9E 10594721 IC50 = 75.3 nM T22939 C8OZH9 10595417 Ki = 5.3 nM T22939 CAYE76 10595774 IC50 = 2000 nM T22939 CBEC38 10596252 Ki = 1.8 nM T22939 C6G7JR 10596379 Ki = 2.6 nM T22939 CX59UV 10596404 EC50 = 124 nM T22939 CC23IP 10596522 Ki = 24.6 nM T22939 C4T7YN 10597442 Ki > 500 nM T22939 CU0IQ6 10598087 Ki = 2.4 nM T22939 CTP6N9 10598088 Ki = 0.93 nM T22939 CC8T7J 10598305 Ki = 3.4 nM T22939 CGQK63 10610968 IC50 = 109 nM T22939 C0UWZ7 10613134 Ki = 10 nM T22939 CEI98J 10614884 IC50 = 543 nM T22939 C3W1BN 10615956 IC50 = 274 nM T22939 CBJ8N5 10615957 IC50 = 2708 nM T22939 CXUS14 10615958 IC50 = 585 nM T22939 CAD6L2 10618033 Ki = 22 nM T22939 CT1M6R 10618939 IC50 = 270 nM T22939 CMK8I6 10622122 Ki = 0.48 nM T22939 CO3V0S 10622594 Ki = 0.55 nM T22939 C6NR3F 10623146 Ki = 8.7 nM T22939 CM1LK7 10639438 IC50 > 1000 nM T22939 C1U0KY 10640594 IC50 = 136 nM T22939 CKO58S 10641642 IC50 = 48.2 nM T22939 C2KD6N 10643454 Ki = 70 nM T22939 C57PFY 10643931 EC50 = 8.7 nM T22939 C02ZMG 10643956 Ki = 0.43 nM T22939 C21WAD 10644405 Ki = 8.8 nM T22939 CZ13MS 10644734 Ki = 31.3 nM T22939 CXK76H 10645656 Ki = 5.3 nM T22939 CF08PC 10661117 Ki = 119 nM T22939 C97HTI 10662571 IC50 = 49 nM T22939 C1RIM7 10662717 IC50 = 348 nM T22939 C3RTS7 10663608 IC50 = 3346 nM T22939 C4B0WQ 10665308 IC50 = 98 nM T22939 CU9X3A 10665612 Ki = 31 nM T22939 CEOX63 10667091 Ki = 10.5 nM T22939 C69CNF 10667548 Ki = 4.9 nM T22939 CL0O4M 10668663 Ki = 18.7 nM T22939 CYNG45 10668755 Ki = 1.5 nM T22939 CS5QI9 10683040 IC50 > 1000 nM T22939 C72FRC 10688714 IC50 > 1000 nM T22939 CS6YF0 10690456 Ki = 6.6 nM T22939 CYRQ10 10691647 Ki = 0.74 nM T22939 CA8FU6 10691738 IC50 > 1000 nM T22939 C6SP3O 10694256 EC50 = 14 nM T22939 CZM1G3 10710737 IC50 > 1000 nM T22939 CY81CQ 10710954 IC50 = 1678 nM T22939 C1Q0BO 10710955 IC50 > 10000 nM T22939 CP7G8A 10711095 IC50 = 3726 nM T22939 CVD2Y9 10717098 Ki = 1.7 nM T22939 CK2NM9 10717832 EC50 = 16 nM T22939 CIU2Q7 10733732 IC50 = 1239 nM T22939 CG3MQ7 10734760 IC50 = 3277 nM T22939 C1MA4E 10735732 IC50 = 3162 nM T22939 CYG5F4 10738747 Ki = 13.3 nM T22939 CUG2Z9 10739308 Ki = 59.6 nM T22939 CJ3HF2 10739813 Ki = 2.7 nM T22939 CAT1X8 10741366 Ki = 1.1 nM T22939 C26DFK 10741917 Ki = 5.5 nM T22939 C3H6CZ 10754393 Ki = 88 nM T22939 CBHG38 10758309 IC50 = 735 nM T22939 C0VSE9 10759031 IC50 = 170 nM T22939 CRF6B3 10759291 IC50 = 398 nM T22939 CX2F8U 10763495 Ki = 60 nM T22939 CF57BT 10763575 EC50 = 22 nM T22939 CB3JD0 10763832 Ki = 0.41 nM T22939 C0NB2H 10765513 Ki = 0.78 nM T22939 C3XBT9 10780550 IC50 = 515 nM T22939 CJ4D6M 10782071 IC50 = 393 nM T22939 CEC5Z2 10782232 IC50 = 310 nM T22939 C7HAB1 10782276 Ki = 441 nM T22939 CNV27D 10783127 Ki = 156 nM T22939 C7EF4Q 10783200 IC50 = 1105 nM T22939 CNL1U7 10785305 Ki = 275 nM T22939 CXG39T 10786881 Ki = 53.3 nM T22939 C6VSY3 10787222 Ki = 24.3 nM T22939 C07BOR 10787258 Ki = 1.2 nM T22939 CF84OK 10805052 Ki = 5 nM T22939 C10AMX 10805958 Ki = 69 nM T22939 C35YZT 10806774 IC50 = 1828 nM T22939 CBX48C 10807828 Ki = 109 nM T22939 CN5WV4 10809583 Ki = 84 nM T22939 CUB74K 10810135 Ki = 0.37 nM T22939 CN42SF 10810393 Ki = 10.1 nM T22939 C1CRQ5 10811045 Ki = 3.6 nM T22939 C6O0TN 10812672 Ki = 13.8 nM T22939 C2AH8G 10812960 Ki = 6.8 nM T22939 C2IX6J 10813169 Ki = 22.1 nM T22939 C0U7OX 10825740 Ki = 181.97 nM T22939 CL7JN6 10827013 Ki = 28.8 nM T22939 C4NWT7 10829815 IC50 = 2334 nM T22939 CGDE16 10830327 IC50 > 1000 nM T22939 CD4G1K 10830667 IC50 = 1763 nM T22939 CR42IT 10831262 IC50 = 270 nM T22939 CN1H5Z 10832792 Ki = 2.3 nM T22939 CV53LK 10833845 Ki = 3.5 nM T22939 C2WHK5 10834892 Ki = 12.6 nM T22939 CL6R3O 10835889 Ki = 1.3 nM T22939 CEX18K 10836526 Ki = 3.9 nM T22939 CC20YZ 10837490 Ki = 1.1 nM T22939 CYRE47 10851308 IC50 = 390 nM T22939 CP4K9Q 10853414 IC50 = 876 nM T22939 CTF24A 10854079 IC50 = 4000 nM T22939 CX68SV 10854490 IC50 = 2931 nM T22939 CA96PR 10860931 Ki = 2920 nM T22939 CHU9A4 10873317 EC50 = 2 nM T22939 CI5F0S 10881662 Ki = 4.8 nM T22939 CVG34R 10883247 Ki = 450 nM T22939 CK41RM 10892050 Ki > 10000 nM T22939 C2T0YG 10895941 Ki = 6.4 nM T22939 CP9FX4 10904951 Ki > 5000 nM T22939 C54IAT 10905085 Ki > 5000 nM T22939 C6EG2D 10906030 Ki = 34 nM T22939 CBD12K 10906044 Ki = 1.2 nM T22939 CNL4U1 10916564 EC50 = 11 nM T22939 C2UG0A 10937849 Ki = 0.62 nM T22939 CLZX29 10938818 Ki = 1.6 nM T22939 CFY3J5 10949008 Ki = 1.5 nM T22939 CHU10G 10960295 EC50 = 1.4 nM T22939 CT2BR8 10969959 Ki = 435 nM T22939 C0GX6P 10970905 Ki = 966 nM T22939 CV3QY8 10972344 Ki = 22 nM T22939 CA4EM2 10982273 Ki = 0.62 nM T22939 CWZ58Y 10982496 Ki = 2.6 nM T22939 CY4U5J 10990453 EC50 = 75 nM T22939 CJ8SM3 10993078 EC50 = 2.7 nM T22939 C07JFA 10993685 Ki = 0.59 nM T22939 CUC05J 11002535 Ki = 192 nM T22939 C8AY9Z 11003946 Ki = 3080 nM T22939 CMJ7F9 11013871 Ki > 5000 nM T22939 C7E9XI 11015162 EC50 = 0.93 nM T22939 CY6IV2 11023208 Ki = 6.1 nM T22939 CRH3L8 11025398 Ki = 0.61 nM T22939 C2RE3P 11037903 EC50 = 9 nM T22939 CU02DM 11046701 Ki = 4740 nM T22939 CZ26AF 11047249 Ki = 9.2 nM T22939 CUYB81 11057924 Ki = 100 nM T22939 CZPG50 11058826 EC50 = 12 nM T22939 CIH8K4 11066740 Ki > 10000 nM T22939 C53JVG 11069432 Ki = 0.71 nM T22939 CS7Q4F 11069511 Ki = 200 nM T22939 CI8GJ5 11079263 EC50 = 1.7 nM T22939 C09ZLY 11088436 Ki > 10000 nM T22939 C6T7CR 11089159 Ki = 1460 nM T22939 C6HPL0 11089468 Ki = 61 nM T22939 C6LYG7 11090322 Ki = 2.089 nM T22939 CE2O8Y 11110616 Ki = 2400 nM T22939 C69GXQ 11110815 Ki = 2100 nM T22939 CJNP35 11112717 Ki = 1.9 nM T22939 CDX2W3 11121575 Ki = 730 nM T22939 C1OJK3 11131414 Ki = 330 nM T22939 CBDG76 11132271 Ki > 5000 nM T22939 C6TJ8D 11132273 Ki = 200 nM T22939 C1W0RZ 11152632 IC50 = 54.4 nM T22939 CA5IX8 11153117 IC50 = 30 nM T22939 CXS6J7 11155441 Ki = 190 nM T22939 C1G5VI 11161470 EC50 = 245.8 nM T22939 C5C7OM 11175557 IC50 = 100 nM T22939 CDT7J9 11176296 IC50 = 1000 nM T22939 CE1G5Z 11176845 IC50 = 66.1 nM T22939 C2RCO3 11187174 EC50 = 0.5 nM T22939 C3LSZ6 11187938 IC50 = 8.4 nM T22939 C1QCP5 11198503 IC50 = 205.8 nM T22939 CP3D7X 11201812 IC50 > 2000 nM T22939 CGB6E3 11210694 EC50 = 0.8 nM T22939 CL97OU 11212803 IC50 = 1210 nM T22939 C4U0DF 11213029 Ki = 1400 nM T22939 C7CP4Z 11221807 EC50 = 1.1 nM T22939 C6K5WD 11223971 IC50 = 78.2 nM T22939 CLCM91 11224044 Ki = 400 nM T22939 CF3AY1 11225369 IC50 > 2000 nM T22939 CRN4V2 11232136 IC50 = 25 nM T22939 CHI2R9 11233809 IC50 = 9 nM T22939 CUOW53 11234644 IC50 = 1000 nM T22939 CB9NC5 11246330 IC50 = 59.2 nM T22939 CYCR06 11256303 IC50 > 1000 nM T22939 C1VHT8 11257462 IC50 = 8.1 nM T22939 CG80FU 11257463 IC50 = 5 nM T22939 CY5C7N 11258139 IC50 = 116.7 nM T22939 C8XPZ4 11269445 IC50 > 2000 nM T22939 C4HNB8 11269886 IC50 > 2000 nM T22939 CJLC62 11273833 IC50 = 140 nM T22939 CC0XI4 11279959 EC50 = 0.8 nM T22939 C4SC0W 11281576 IC50 > 1000 nM T22939 C8YL6K 11282486 IC50 > 2000 nM T22939 CUX0S2 11282904 Ki = 790 nM T22939 CIY9H5 11291999 IC50 > 2000 nM T22939 CZW24E 11292160 IC50 = 65.5 nM T22939 C0IQ9K 11304445 IC50 = 1450 nM T22939 C0XUF2 11305564 IC50 > 1000 nM T22939 CB1IL8 11306419 EC50 = 0.2 nM T22939 CYOD61 11314184 IC50 = 14.5 nM T22939 C40JLN 11315741 IC50 = 138.3 nM T22939 C9TH6D 11316707 IC50 = 10 nM T22939 C9N6OY 11324250 IC50 = 3.3 nM T22939 CFM3N6 11325538 EC50 = 0.7 nM T22939 C0B2FT 11327284 IC50 = 240 nM T22939 CXC9G3 11327341 IC50 > 2000 nM T22939 C1HZS7 11336351 IC50 > 1000 nM T22939 CT9Y4O 11339440 IC50 = 11.3 nM T22939 CS2LZ7 11360922 EC50 = 37.5 nM T22939 CWH2G5 11361328 IC50 = 56.6 nM T22939 CP2DL0 11377050 IC50 = 150 nM T22939 C76VYN 11382721 IC50 > 2000 nM T22939 CV4RO2 11384310 IC50 = 200 nM T22939 CXW40M 11384346 IC50 > 2000 nM T22939 CQ8CB6 11393997 IC50 = 56 nM T22939 C0K1QX 11403275 EC50 = 137.7 nM T22939 CD4O3M 11404458 EC50 = 30.5 nM T22939 CU7IE0 11410199 IC50 = 1700 nM T22939 CO20QH 11416730 EC50 = 0.4 nM T22939 C1KG4U 11417145 IC50 = 42.2 nM T22939 C5WO0U 11429662 IC50 > 1000 nM T22939 C6KNX4 11440728 IC50 = 119.8 nM T22939 CNVX52 11464170 IC50 = 349.4 nM T22939 CK61QZ 11464996 IC50 = 26.6 nM T22939 CU9GM7 11474806 IC50 = 36.5 nM T22939 CD2Q3F 11474917 IC50 = 490 nM T22939 CC75NQ 11477616 Ki = 840 nM T22939 CQ62KS 11485693 IC50 = 11.8 nM T22939 C3HBD9 11486844 IC50 = 365.7 nM T22939 C2JC5K 11493567 IC50 = 13 nM T22939 C9Q1NY 11494167 Ki = 75 nM T22939 CFLQ08 11495227 IC50 > 2000 nM T22939 C03NYX 11495549 IC50 = 6000 nM T22939 C9V7PD 11500344 IC50 = 15 nM T22939 CFH92S 11500731 IC50 = 30 nM T22939 C0O7TM 11500993 Ki = 370 nM T22939 CC16NH 11515319 IC50 = 4.5 nM T22939 CR40IH 11516847 IC50 = 1800 nM T22939 C4Q5XE 11517391 Ki = 420 nM T22939 CP4F8X 11517412 IC50 = 450 nM T22939 C1R6DC 11531942 IC50 > 2000 nM T22939 CZ1HA3 11538472 IC50 > 2000 nM T22939 CFC1Z4 11538799 IC50 > 2000 nM T22939 CX8BO4 11543708 IC50 = 4.7 nM T22939 CI90JB 11551816 Ki = 450 nM T22939 C0J8UL 11551817 Ki = 230 nM T22939 CH2KP9 11555183 IC50 = 0.61 nM T22939 CBK60G 11559947 IC50 = 8 nM T22939 C1D9YS 11560003 IC50 > 2000 nM T22939 CB37YF 11566981 Ki = 151 nM T22939 C5UEY6 11567352 Ki = 25 nM T22939 C8WJ2F 11567609 IC50 = 130 nM T22939 CY7DV1 11574319 IC50 = 164 nM T22939 CZ68MI 11574590 IC50 = 351 nM T22939 C0SCT6 11588584 IC50 = 190 nM T22939 C3MW1D 11589982 IC50 = 1300 nM T22939 C03QYZ 11590471 IC50 = 750 nM T22939 CZO0L1 11595527 Ki = 70 nM T22939 CAO2P1 11596392 IC50 > 2000 nM T22939 CD5T0O 11608377 IC50 = 20 nM T22939 C7YS3I 11609033 IC50 > 10000 nM T22939 CCYP20 11616167 IC50 = 5.5 nM T22939 CSB97O 11617028 Ki = 8.2 nM T22939 CC49FR 11617298 Ki = 650 nM T22939 CR5DA0 11617684 Ki = 650 nM T22939 CA2D1P 11624781 IC50 = 194 nM T22939 C3P6BI 11631677 IC50 = 25 nM T22939 CRF4E1 11631740 Ki = 1400 nM T22939 CW6R3T 11631784 Ki = 15 nM T22939 CRL3A7 11632925 IC50 = 2400 nM T22939 CQB0E3 11633482 IC50 = 530 nM T22939 C2Z6QV 11634852 Ki < 3162.28 nM T22939 C3B1YP 11638175 IC50 = 29 nM T22939 CKYE81 11638660 IC50 = 30 nM T22939 C9DNG1 11640164 IC50 > 2000 nM T22939 CB4E0S 11645780 Ki = 2300 nM T22939 C3MHY7 11646048 Ki = 22 nM T22939 C1RJ3I 11646689 IC50 > 2000 nM T22939 CX3L5S 11647533 IC50 > 2000 nM T22939 CU3K9V 11653520 Ki = 14 nM T22939 C4S5RG 11655053 IC50 > 2000 nM T22939 CWXF31 11659518 IC50 = 5.6 nM T22939 CDOZ32 11661172 IC50 = 1900 nM T22939 C0LEZ3 11667800 Ki = 1300 nM T22939 C5XEN0 11668719 IC50 > 10000 nM T22939 CEC7P6 11673811 IC50 > 10000 nM T22939 CX6O8C 11673997 IC50 = 4.9 nM T22939 CM57PA 11682250 Ki = 520 nM T22939 CZPK72 11682989 IC50 = 3600 nM T22939 C8SY4D 11688929 Ki = 1400 nM T22939 CCK83U 11690269 IC50 = 160 nM T22939 CY07JH 11696378 IC50 > 2000 nM T22939 CBU02W 11696959 IC50 = 790 nM T22939 C2S9IT 11697271 IC50 > 2000 nM T22939 CGR32I 11697882 IC50 = 1700 nM T22939 C42NIT 11697950 Ki = 270 nM T22939 CPA26L 11701694 IC50 = 10 nM T22939 C89AFS 11702581 IC50 = 27 nM T22939 C3OQH4 11703401 Ki = 6600 nM T22939 C75IBX 11704529 IC50 = 5900 nM T22939 CGX54N 11704756 IC50 > 10000 nM T22939 CO2N1W 11710364 IC50 > 2000 nM T22939 C8OPA1 11710962 IC50 > 2000 nM T22939 C1WO7R 11711144 Ki = 19.95 nM T22939 CW3N8H 11711766 IC50 = 2000 nM T22939 COEU05 11719039 IC50 = 700 nM T22939 C6KW3Z 11722813 EC50 = 200 nM T22939 C6HGB2 11722878 EC50 = 2.5 nM T22939 C9DK4N 11723766 IC50 = 100 nM T22939 CM3BG2 11724520 IC50 > 2000 nM T22939 CID9O5 11726380 EC50 = 5.7 nM T22939 C4OH1Y 11726899 Ki > 10000 nM T22939 C0VJ3I 11727825 Ki > 5000 nM T22939 CVA1S3 11728656 Ki = 29 nM T22939 CZ0B7H 11731863 EC50 = 0.71 nM T22939 CUJ2R1 11733088 EC50 = 14 nM T22939 CR12UX 11738282 IC50 = 1660 nM T22939 CPN1X7 11739446 IC50 = 13.1 nM T22939 C57WMZ 11739563 EC50 = 110 nM T22939 CQO76Z 11741168 IC50 > 2000 nM T22939 C87YNC 11741891 IC50 = 240 nM T22939 CH92VI 11743259 IC50 = 640 nM T22939 CQI39V 11749248 IC50 = 14.6 nM T22939 CY74EX 11749286 IC50 = 29.8 nM T22939 CM89PZ 11749484 IC50 = 62.5 nM T22939 CVD63Y 11749908 IC50 = 32.2 nM T22939 C5HLU8 11750204 IC50 = 1150 nM T22939 CY1F4I 11752649 Ki = 1780 nM T22939 CKD9R8 11757239 IC50 = 47 nM T22939 CQU0E7 11774868 IC50 = 395 nM T22939 COI0P1 11774981 IC50 > 2000 nM T22939 CR70FP 11794088 Ki = 21 nM T22939 C18XFI 11795355 Ki = 0.55 nM T22939 CXDP07 11798449 Ki = 0.59 nM T22939 CU7EJ1 11822858 Ki > 10000 nM T22939 C5FRJ6 11825145 Ki = 390 nM T22939 C7G3CH 12042978 IC50 = 56 nM T22939 CGR38Y 12043185 EC50 = 1.05 nM T22939 C4U8KY 12085089 IC50 = 367 nM T22939 CBMH81 14001634 IC50 = 510 nM T22939 CB7Q3A 15440425 Ki = 66 nM T22939 C0LE3M 15458731 Ki = 12.88 nM T22939 CF4O7Z 15458732 Ki = 199.53 nM T22939 C1G9EX 15458733 Ki = 15.49 nM T22939 C5U6ZV 15458734 Ki = 23.99 nM T22939 CXIR52 15458735 Ki = 181.97 nM T22939 C8BZJ0 15458736 Ki = 77 nM T22939 C7FA1K 15458737 Ki = 2.291 nM T22939 C36IOD 15458738 Ki = 12.3 nM T22939 C20ZJY 15458739 Ki = 28.84 nM T22939 C2S1UF 15458740 Ki = 3.467 nM T22939 CJ8C0A 15458741 IC50 = 164 nM T22939 CK5JY2 15458742 Ki = 57 nM T22939 CW40IA 15458746 IC50 = 59 nM T22939 CQ08MF 15458747 Ki = 169 nM T22939 C14LTD 15463551 IC50 = 15.85 nM T22939 C8FVY9 15604499 IC50 = 1.5 nM T22939 C01QWU 16004659 EC50 = 19 nM T22939 CMLY25 16004661 EC50 = 10 nM T22939 CU7H9K 16037461 IC50 = 167 nM T22939 CXT83S 16037462 IC50 = 76 nM T22939 CB8T7N 16037463 IC50 = 78 nM T22939 CS53LY 16037464 IC50 = 75 nM T22939 C92FRI 16037744 Ki = 25.12 nM T22939 C98XWA 16050901 IC50 = 10 nM T22939 C0UG3P 16050904 IC50 = 58 nM T22939 CNI38X 16051001 IC50 = 9 nM T22939 C7Q4TK 16051002 IC50 = 8 nM T22939 CW95VN 16051004 IC50 = 30 nM T22939 CB1L8K 16051005 IC50 = 6 nM T22939 COR4M2 16051097 IC50 = 57 nM T22939 CBV90A 16051102 IC50 = 12 nM T22939 CU7IA9 16051188 IC50 = 36 nM T22939 C9QTK1 16051279 IC50 = 128 nM T22939 C8P5XQ 16051281 IC50 > 3000 nM T22939 CMZH47 16051364 IC50 = 11.7 nM T22939 CA4W5P 16051367 IC50 = 8 nM T22939 C3QOV0 16099227 IC50 > 2000 nM T22939 CW6LO1 16099229 IC50 > 2000 nM T22939 C2R4PK 16099231 IC50 > 2000 nM T22939 C9KM7X 16099232 IC50 > 2000 nM T22939 C05CYN 16099234 IC50 > 2000 nM T22939 CJQ8A1 16099236 IC50 = 555 nM T22939 CA72YW 16099237 IC50 > 2000 nM T22939 CS07DB 16099238 IC50 = 48 nM T22939 C42ESN 16099240 IC50 = 960 nM T22939 CMZ91J 16099242 IC50 > 2000 nM T22939 CF69RC 16099243 IC50 > 2000 nM T22939 C60GEM 16099245 IC50 > 2000 nM T22939 CE48CS 16099246 IC50 > 2000 nM T22939 CTF2M7 16099247 IC50 = 90 nM T22939 CX9BK2 16099248 IC50 > 2000 nM T22939 CN6PA9 16099249 IC50 = 106 nM T22939 C9Z6AK 16099250 IC50 = 240 nM T22939 C5Z8HR 16099251 IC50 = 525 nM T22939 CWK76M 16099252 IC50 = 340 nM T22939 CC24LB 16110489 EC50 > 10 nM T22939 C3RVJ2 16119194 IC50 = 6 nM T22939 CY7O0I 16119239 IC50 = 10 nM T22939 CD6M9L 16119240 IC50 = 35 nM T22939 C8ZH6A 16119245 IC50 = 7 nM T22939 C3BU9M 16216822 IC50 = 1200 nM T22939 C1Q5SV 16220168 IC50 > 10000 nM T22939 C9Z3PU 16225747 IC50 = 28 nM T22939 CH6CN0 16658901 Ki = 2800 nM T22939 CIBY49 16661548 EC50 = 25 nM T22939 C45KPZ 16661549 EC50 = 1 nM T22939 CH60SU 16661701 IC50 = 20 nM T22939 CU9LS2 16661702 EC50 = 3 nM T22939 C1UY8J 16666386 IC50 = 770 nM T22939 C0Y2OK 16721017 IC50 = 1.4 nM T22939 CE71BC 16722203 IC50 = 0.27 nM T22939 CF6V2J 16730097 IC50 = 0.75 nM T22939 CWK35C 16730429 IC50 = 2500 nM T22939 CLC2Z8 16739323 IC50 = 7.5 nM T22939 CSKX58 17758233 Ki = 2290 nM T22939 C7CPW9 17758234 Ki = 38 nM T22939 CI5KT6 17758236 Ki = 57 nM T22939 CK4UP0 17921928 Ki = 273 nM T22939 CG7SZ2 17921931 Ki = 85.11 nM T22939 C8A0FW 17921932 Ki = 44.67 nM T22939 C3FP7L 17921933 Ki = 6.1 nM T22939 CX03YG 18188955 IC50 = 210 nM T22939 CRTO81 18374557 EC50 = 8.2 nM T22939 CKE7O0 18374561 EC50 = 10.9 nM T22939 CR19ST 18512166 IC50 = 7600 nM T22939 CEN14G 18512334 IC50 = 790 nM T22939 CS9CI5 18551230 IC50 = 16 nM T22939 CBI64N 18551237 IC50 = 12.59 nM T22939 CLUA26 18551266 IC50 = 85 nM T22939 C5ZYJ0 20231824 Ki = 104 nM T22939 CEH7V5 20786216 IC50 > 1000 nM T22939 CF0S6J 21210483 IC50 = 33 nM T22939 C40TDI 21210578 IC50 = 410 nM T22939 C1FJU8 21824365 IC50 = 7100 nM T22939 C97WCO 21941658 IC50 = 7.943 nM T22939 CCI89R 21948853 IC50 > 1000 nM T22939 CB2SF4 21948904 IC50 > 1000 nM T22939 C3V9UW 21986241 IC50 = 29 nM T22939 CIN4J2 21986251 EC50 = 2.3 nM T22939 CEJT23 21986260 IC50 = 13.6 nM T22939 CE9G1L 21986274 IC50 = 267 nM T22939 CF6GR4 22019345 IC50 = 38 nM T22939 C04YBK 22019347 IC50 = 13 nM T22939 C8O1UI 22019348 IC50 = 36 nM T22939 C5AH6M 22019349 IC50 = 20 nM T22939 C8LYE4 22019363 IC50 = 28 nM T22939 C5THV1 22019384 IC50 = 29 nM T22939 CY95CQ 22038447 Ki = 38.4 nM T22939 C2ZP7V 22218142 IC50 = 570 nM T22939 CWA9Q6 22284899 IC50 = 400 nM T22939 C1QTK4 22398492 IC50 = 145 nM T22939 C6CSB4 22398502 IC50 > 2000 nM T22939 CR8N1E 22398506 IC50 > 2000 nM T22939 CM83TU 22398533 IC50 = 255 nM T22939 C34LHW 22398559 IC50 > 2000 nM T22939 CJBW90 22398592 IC50 > 2000 nM T22939 CEJ65O 22398627 IC50 = 815 nM T22939 CCYS56 22566499 IC50 > 2000 nM T22939 CGE03P 22566506 IC50 > 2000 nM T22939 CH29BV 22566507 IC50 = 600 nM T22939 C21YKI 22566509 IC50 > 2000 nM T22939 CU8D7L 22566515 IC50 > 2000 nM T22939 C7YMV6 22774896 IC50 = 1600 nM T22939 COY32J 23003206 IC50 = 36 nM T22939 C0QW6U 23041743 Ki = 14 nM T22939 CE9OR4 23433451 Ki = 25 nM T22939 CYR3I6 23433462 IC50 = 353 nM T22939 C0K6ZJ 23433498 Ki = 12 nM T22939 C6UZD7 23433503 Ki = 2.57 nM T22939 CGY94Z 23433542 IC50 = 27 nM T22939 C84MWR 23433579 Ki = 3.6 nM T22939 CQ7X4E 23433633 IC50 = 365 nM T22939 C2T0KG 23433647 Ki = 28.84 nM T22939 C1EOP3 23433683 EC50 = 71 nM T22939 CE82ZP 23435578 EC50 = 0.35 nM T22939 CXNG28 23435580 EC50 = 0.8 nM T22939 CY8GW5 23435581 EC50 = 4.55 nM T22939 C35XIV 23435583 EC50 = 0.9 nM T22939 CG1Z6T 23435587 EC50 = 1.7 nM T22939 CFJ32R 23435589 EC50 = 0.2 nM T22939 CU4F1G 23435590 EC50 = 32 nM T22939 C35HWF 23435593 EC50 = 9.2 nM T22939 C6RD4J 23435594 IC50 = 2087 nM T22939 CI6GZ7 23435595 EC50 = 2.6 nM T22939 CX2FT5 23435602 EC50 = 2.9 nM T22939 CDT63J 23435603 EC50 = 2.4 nM T22939 CD0FR5 23435611 EC50 = 2.4 nM T22939 C6XI4U 23435613 EC50 = 3.5 nM T22939 CU2Z0C 23435614 EC50 = 23 nM T22939 C9O6RB 23596322 Ki > 10000 nM T22939 CF4UA3 23648072 IC50 = 540 nM T22939 C1XA3Y 23727880 IC50 = 78 nM T22939 CWPH96 24180508 EC50 = 0.1 nM T22939 CZ9N1A 24180647 IC50 = 4450 nM T22939 CZI4C6 24739672 Ki = 0.32 nM T22939 CS23KY 24739834 Ki = 1.45 nM T22939 C1M9QG 24739836 Ki = 4.23 nM T22939 CG5SJ0 24739997 Ki = 0.795 nM T22939 C7Z1HW 24740156 Ki = 0.834 nM T22939 CTE1N2 24748569 EC50 > 10000 nM T22939 C4WYE7 24749678 Ki = 137 nM T22939 CY2JS4 24749684 Ki = 1230 nM T22939 C2QHO3 24749808 Ki = 162.9 nM T22939 C6YB7N 24758659 IC50 = 27.4 nM T22939 C0EKO1 24758661 IC50 = 9.2 nM T22939 CR1G7M 24768971 EC50 = 794.33 nM T22939 C5S6JN 24780149 IC50 > 1000 nM T22939 CW5TJ7 24781731 IC50 > 1000 nM T22939 C8F7WP 24811980 IC50 = 8800 nM T22939 CGY0S6 24824069 IC50 = 3.3 nM T22939 CTNY64 24824070 IC50 = 20.3 nM T22939 CGT1C9 24824071 IC50 = 3.2 nM T22939 CR28EY 24824334 IC50 = 30 nM T22939 C35JSL 24824469 EC50 = 1.3 nM T22939 CNM45B 24850992 IC50 = 520 nM T22939 C1JTW2 24851053 Ki = 6.17 nM T22939 CC53XL 24860583 Ki = 1479 nM T22939 C9RLM8 24865155 IC50 = 180 nM T22939 C58NZJ 24865524 Ki = 6.7 nM T22939 CGE0V4 24882669 IC50 > 10000 nM T22939 C58RHY 24883011 IC50 = 4900 nM T22939 CW35CK 24883012 IC50 = 1800 nM T22939 C3SC0V 24883054 IC50 = 1800 nM T22939 C4SA6C 24883055 IC50 = 2400 nM T22939 C2H6BU 24895095 EC50 = 5.4 nM T22939 C5LZK2 24895096 EC50 = 0.5 nM T22939 C19PKU 24895098 EC50 = 0.4 nM T22939 CA7XS2 24895099 EC50 = 3.4 nM T22939 COGP96 24936313 Ki > 5000 nM T22939 CVY09S 24936449 Ki = 406 nM T22939 CBN24H 24936982 Ki = 109 nM T22939 C06PDG 24952192 Ki = 22 nM T22939 CG1CF9 24952193 Ki = 53 nM T22939 CZC7L8 24953162 IC50 = 1160 nM T22939 C4W7BN 24954947 IC50 = 790 nM T22939 C6XC2R 24954951 IC50 > 12000 nM T22939 C50XFU 24956011 IC50 = 100 nM T22939 C50EAQ 24956012 IC50 = 62.1 nM T22939 C5COZ7 24956013 IC50 = 29.3 nM T22939 CK67LB 24956014 IC50 = 29.1 nM T22939 C26ITJ 24956015 IC50 = 15.7 nM T22939 C6E7FV 24956376 IC50 = 15 nM T22939 C0FQC5 24956377 IC50 = 34.6 nM T22939 C2KUT4 24956729 EC50 = 3.3 nM T22939 C1Q2RA 24956731 IC50 = 30 nM T22939 CI83HO 24956732 EC50 = 35.8 nM T22939 CF5CK7 24957093 IC50 = 30.1 nM T22939 CPN6Y8 24957094 IC50 = 14.9 nM T22939 CYES17 24957737 Ki = 2269 nM T22939 C83YKB 24961057 Ki > 1250 nM T22939 CIGM27 24983460 IC50 = 2000 nM T22939 CJM73Y 24987018 IC50 = 34 nM T22939 C8OZ3H 24987026 IC50 = 800 nM T22939 CO30YU 24987374 IC50 = 115 nM T22939 CCF34H 24987375 IC50 = 266 nM T22939 CFI8D1 24987376 IC50 = 300 nM T22939 C0LIQ3 24987377 IC50 = 3 nM T22939 C14EFU 24990122 IC50 = 20 nM T22939 C80LEK 24990485 IC50 = 63 nM T22939 CMD98H 24990837 IC50 = 79 nM T22939 CNMD47 24990839 IC50 = 50 nM T22939 CHY0D7 25013322 IC50 = 910 nM T22939 C0TPS5 25013653 IC50 > 10000 nM T22939 CWU91M 25013811 IC50 > 20000 nM T22939 CSH29L 25013812 IC50 = 630 nM T22939 C2G1JK 25053351 Ki > 30000 nM T22939 CXKF32 25066493 IC50 = 4070 nM T22939 CAW8M0 25070694 IC50 = 28.4 nM T22939 CWUA34 25093229 IC50 > 10000 nM T22939 C67SAZ 25110681 EC50 = 3 nM T22939 C0PTE9 25110682 EC50 = 0.81 nM T22939 C3XNB2 25110683 EC50 = 0.96 nM T22939 CZDE94 25110695 EC50 = 1.3 nM T22939 CF1S8P 25132150 IC50 = 340 nM T22939 CB56QH 25132505 IC50 = 780 nM T22939 C35HKY 25145080 Ki = 236 nM T22939 CXF9G0 25145082 Ki = 23 nM T22939 C21XDY 25145083 Ki = 54 nM T22939 CANT87 25145217 Ki = 39 nM T22939 CE1I7A 25145499 Ki = 574 nM T22939 CV6N1P 25145500 Ki = 8.5 nM T22939 CS6JQ1 25167502 Ki = 1400 nM T22939 C0XPW9 25168896 IC50 = 6400 nM T22939 CUL27D 25168900 IC50 = 3200 nM T22939 CEV2D7 25205475 IC50 = 5000 nM T22939 C9S0ZW 25205477 IC50 = 1500 nM T22939 C49KHR 25206116 IC50 > 10000 nM T22939 CNQ9Y0 25231294 IC50 = 0.25 nM T22939 CVL47Y 25231295 IC50 = 0.17 nM T22939 C87ZHT 25231296 IC50 = 0.095 nM T22939 C5I3ZH 25231297 IC50 = 0.025 nM T22939 C6GSB2 25231472 IC50 = 0.38 nM T22939 C8KZ0B 25231473 IC50 = 0.073 nM T22939 CHM49K 25231474 IC50 = 34 nM T22939 CAON04 25231475 IC50 = 0.27 nM T22939 C1MWA2 25231476 IC50 = 0.16 nM T22939 CTPB29 25231634 IC50 = 0.63 nM T22939 C5DQY1 25231635 IC50 = 0.9 nM T22939 C5Z1PU 25231636 IC50 = 100 nM T22939 CAD2V4 25231637 IC50 = 1.8 nM T22939 C8HB6E 25231806 IC50 = 0.73 nM T22939 C9OG3W 25231807 IC50 = 0.16 nM T22939 CP0R1E 25231808 IC50 = 2.2 nM T22939 C7CK8P 25231809 IC50 = 0.44 nM T22939 C4LI5T 25231979 IC50 = 2.1 nM T22939 CNOJ86 25231980 IC50 = 1.2 nM T22939 CCWB43 25233236 IC50 = 1 nM T22939 CHG70Z 25233237 IC50 = 0.18 nM T22939 C58ZUA 25233401 IC50 = 0.12 nM T22939 CLZ6F0 25233402 IC50 = 0.071 nM T22939 CR4E5A 25233403 IC50 = 0.15 nM T22939 CH04QJ 25233404 IC50 = 0.44 nM T22939 C93EIC 25233405 IC50 = 0.46 nM T22939 CGC4X3 25233572 IC50 = 0.4 nM T22939 CS1MX3 25233573 IC50 = 0.47 nM T22939 CU9FO4 25233574 IC50 = 0.55 nM T22939 C4CNQ5 25233575 IC50 = 0.69 nM T22939 CI26BG 25233749 IC50 = 78 nM T22939 CJFX31 25233750 IC50 = 1.55 nM T22939 CUB96G 25233751 IC50 = 0.79 nM T22939 C3IBN6 25233752 IC50 = 0.27 nM T22939 CS84RU 25233937 IC50 = 72 nM T22939 C8GZQ4 25233938 IC50 = 1.7 nM T22939 CLMB86 25233939 IC50 = 72 nM T22939 C6LZE2 25233940 IC50 = 0.46 nM T22939 CLY9W3 25235364 IC50 > 1000 nM T22939 CY6X2V 25258136 IC50 = 2600 nM T22939 CV4Y6N 25258138 IC50 = 1100 nM T22939 CNLS64 25258386 IC50 = 750 nM T22939 C1L0UG 40604675 IC50 = 300 nM T22939 CR4C2X 43320749 IC50 = 6950 nM T22939 CX89HM 44138106 Ki = 31 nM T22939 C91KTD 44186997 EC50 = 4.5 nM T22939 C6DOT1 44186998 EC50 = 4 nM T22939 CXZ35T 44193145 Ki = 160 nM T22939 C2MOF7 44193146 Ki = 213 nM T22939 CWR6X1 44193147 Ki = 93 nM T22939 C3JOW4 44193245 Ki = 662 nM T22939 CXR5O7 44250279 IC50 = 1 nM T22939 C9QED8 44250280 IC50 = 34 nM T22939 CHGI03 44251606 IC50 > 2000 nM T22939 CAU2H0 44251621 EC50 = 0.5 nM T22939 C0OA6M 44264483 IC50 = 280 nM T22939 COCE32 44264569 IC50 = 270 nM T22939 CI0TN2 44264577 IC50 = 100 nM T22939 CXOR54 44264579 IC50 = 106 nM T22939 C01HSQ 44264588 IC50 = 440 nM T22939 CL0BI4 44275158 IC50 = 100 nM T22939 CDS6E2 44275349 IC50 = 114 nM T22939 C1QI4H 44275352 EC50 = 1000 nM T22939 CQS5L7 44275356 EC50 = 1000 nM T22939 CZAH03 44275357 IC50 = 100 nM T22939 C6XWK8 44275364 EC50 > 10000 nM T22939 CEK9N3 44275366 IC50 = 100 nM T22939 C57NZK 44275378 IC50 = 100 nM T22939 C0KBH2 44275720 EC50 > 3000 nM T22939 CHJ42T 44275721 EC50 > 3000 nM T22939 C4NDL8 44275733 EC50 = 9.8 nM T22939 C46VWO 44275773 EC50 = 1.9 nM T22939 CK6M3O 44275941 EC50 = 71.4 nM T22939 CP8OC7 44282950 Ki = 0.44 nM T22939 C6X2IH 44295653 IC50 = 2443 nM T22939 CK4J3H 44305217 Ki = 26 nM T22939 C5BT1G 44305218 Ki = 3.09 nM T22939 C1DBA2 44305237 Ki = 7.943 nM T22939 CRU41I 44305238 EC50 = 48 nM T22939 CQF7U6 44305249 Ki = 44.67 nM T22939 C9KC1G 44305269 Ki > 100 nM T22939 CDB54J 44305270 EC50 = 1.7 nM T22939 CQL9B2 44305514 Ki = 16.6 nM T22939 CYRM52 44305525 Ki > 100 nM T22939 COEK92 44305527 Ki > 100 nM T22939 C0XLN6 44305556 EC50 = 0.15 nM T22939 CHB82F 44305684 Ki = 15 nM T22939 C1UK4M 44305720 Ki = 6.761 nM T22939 CTW67P 44305733 Ki = 12.3 nM T22939 C8FBR0 44305734 Ki > 1000 nM T22939 CEP7J0 44305769 EC50 = 178 nM T22939 CC2O4T 44305801 EC50 = 118 nM T22939 CD7C5E 44305809 EC50 = 40 nM T22939 CH4PU5 44305819 IC50 = 1157 nM T22939 CXN1M7 44305835 Ki > 1000 nM T22939 C7SE3Z 44305843 EC50 = 43 nM T22939 CDXK57 44305874 Ki = 13.49 nM T22939 C6N1AR 44305929 EC50 = 52 nM T22939 C2BDY0 44305930 Ki = 288.4 nM T22939 CGT3E0 44305979 IC50 = 811 nM T22939 C2BWL8 44305980 Ki = 391 nM T22939 C8ZR1T 44305991 Ki = 370 nM T22939 C9U6SZ 44306067 Ki = 5.6 nM T22939 C4I0UH 44306083 EC50 = 193 nM T22939 CCX2B3 44309247 EC50 ~ 1000 nM T22939 C47XJE 44309248 EC50 ~ 1000 nM T22939 CVX0I3 44309412 IC50 ~ 3000 nM T22939 C50ZBH 44309489 IC50 = 41 nM T22939 C1DMI8 44309499 EC50 > 1000 nM T22939 C0WYG1 44309500 EC50 > 1000 nM T22939 C24BCA 44309676 EC50 = 130 nM T22939 CLJ98K 44309924 EC50 > 1000 nM T22939 C6AHS5 44325266 Ki = 483 nM T22939 COA36F 44325268 Ki = 2580 nM T22939 C8E6TS 44325286 Ki = 87 nM T22939 CSID10 44325287 Ki = 77 nM T22939 CMW25P 44325290 IC50 = 46 nM T22939 C7YQ1W 44325291 Ki = 53.1 nM T22939 C61TWJ 44325292 IC50 = 10000 nM T22939 CZ25HP 44325293 Ki > 10000 nM T22939 CPBL70 44325294 Ki > 10000 nM T22939 CM6NW2 44325301 IC50 = 74 nM T22939 C38IEA 44325321 Ki = 97 nM T22939 C3EOF1 44325326 Ki = 20.89 nM T22939 CLNK34 44325373 Ki = 3.09 nM T22939 CX42KH 44325387 Ki = 1.5 nM T22939 C37JEN 44325388 Ki = 11.2 nM T22939 CK0N2V 44325502 IC50 = 662 nM T22939 C36BNE 44325530 Ki = 25.5 nM T22939 CXZR46 44325544 IC50 = 29.2 nM T22939 CA4G5C 44325705 Ki = 1858 nM T22939 C1AX8P 44325706 IC50 = 73.1 nM T22939 C7JBY2 44325708 IC50 = 112.8 nM T22939 CW1N3O 44325716 IC50 = 99 nM T22939 CDQW05 44325717 Ki = 101 nM T22939 CNF7S6 44325757 Ki > 10000 nM T22939 CFY3N7 44325758 IC50 = 3061 nM T22939 C0G5BY 44325768 IC50 > 10000 nM T22939 CSF16T 44341592 Ki = 23 nM T22939 C9Y1MP 44341593 Ki = 3.3 nM T22939 CT62WI 44341706 Ki = 0.87 nM T22939 CO10KF 44341745 Ki = 1.1 nM T22939 CDS5W7 44341746 Ki = 3.2 nM T22939 C9JGS0 44341846 Ki = 26.5 nM T22939 CP0AQ3 44341860 Ki = 3.5 nM T22939 CE62XL 44341871 Ki = 0.95 nM T22939 CIFK12 44341872 Ki = 1.7 nM T22939 CXG8Y5 44341873 Ki = 16.4 nM T22939 C6KSD0 44341876 Ki = 1.2 nM T22939 CP6LV3 44341880 Ki = 2.9 nM T22939 CZT6O9 44341890 Ki = 6 nM T22939 CJRZ82 44341891 Ki = 64 nM T22939 CRIY20 44341919 Ki = 24.3 nM T22939 CT15JC 44342090 Ki = 6.6 nM T22939 CKP23I 44342091 EC50 = 49 nM T22939 C8RQS2 44342092 Ki = 1.5 nM T22939 C9VY0G 44343925 IC50 = 70.7 nM T22939 CS6JG3 44343981 IC50 = 100.1 nM T22939 C9GRH5 44344079 IC50 = 206 nM T22939 CDK63E 44344162 IC50 = 32 nM T22939 CZ1T4S 44344264 IC50 = 185 nM T22939 C9KA8X 44344265 IC50 = 85 nM T22939 CDGP02 44353994 Ki = 0.42 nM T22939 C73CXK 44354006 Ki = 1.4 nM T22939 CHE09P 44354630 Ki = 32 nM T22939 CO3U7R 44354644 Ki = 30.9 nM T22939 C8M3SJ 44354645 Ki = 36 nM T22939 CP48SO 44354661 Ki = 37 nM T22939 CAET94 44354707 Ki = 30.9 nM T22939 C9FT3C 44354756 Ki > 100 nM T22939 C0N3TD 44354884 Ki = 12.3 nM T22939 CPQ2A6 44354885 Ki = 6.2 nM T22939 CM0G1V 44354886 Ki = 25.7 nM T22939 C86OTP 44354901 IC50 = 242 nM T22939 C2GEZ4 44355053 Ki = 234.42 nM T22939 CL6G3Q 44355066 Ki = 3.89 nM T22939 CL1VH6 44355082 Ki = 79.43 nM T22939 C16HRA 44355173 IC50 = 52 nM T22939 CSAU31 44377064 IC50 = 750 nM T22939 C7H9NC 44377081 IC50 = 1000 nM T22939 C60DYH 44377090 IC50 = 170 nM T22939 CVH2R3 44377098 IC50 = 150 nM T22939 CYLI63 44377110 IC50 = 380 nM T22939 CQX39I 44377356 IC50 = 430 nM T22939 C9FJW4 44377382 IC50 = 730 nM T22939 C5HW2V 44378589 IC50 = 92.6 nM T22939 CG0J6Y 44378590 IC50 = 47 nM T22939 CM16EI 44378605 EC50 > 10000 nM T22939 C3JES5 44378688 IC50 = 3042 nM T22939 CIR62Q 44378690 IC50 = 51.2 nM T22939 CRF48X 44378790 IC50 = 158.8 nM T22939 C8Y4RP 44393060 IC50 = 200 nM T22939 CK58MC 44393061 IC50 = 32 nM T22939 CTI0L9 44393062 IC50 = 3.8 nM T22939 C13SYV 44396250 Ki = 1.9 nM T22939 CB1P0S 44396251 Ki = 1.1 nM T22939 CHY1C3 44396271 Ki = 1.2 nM T22939 C29MBI 44396272 Ki = 2.4 nM T22939 C4TQ6N 44396282 Ki = 0.81 nM T22939 CH2Y3L 44396283 Ki = 0.96 nM T22939 CWZB52 44396284 Ki = 3.5 nM T22939 CD80LM 44396296 Ki = 6.4 nM T22939 C6SI5L 44396297 Ki = 0.39 nM T22939 CR4H1E 44396316 Ki = 1 nM T22939 C45LRH 44396317 Ki = 0.53 nM T22939 C5JG6H 44396330 Ki = 2.1 nM T22939 CA8V4G 44396331 Ki = 4.4 nM T22939 C57CPQ 44396332 Ki = 4.6 nM T22939 CM29RA 44397719 IC50 = 11.7 nM T22939 C5LN4G 44397730 IC50 = 29 nM T22939 CDLB25 44397734 IC50 = 412.3 nM T22939 CV60LH 44397751 IC50 = 77.9 nM T22939 C3TH9F 44397754 IC50 = 96.8 nM T22939 CFUK82 44397777 IC50 = 134.7 nM T22939 C9G8FO 44397790 IC50 = 105.6 nM T22939 CB73AI 44397804 IC50 = 60.3 nM T22939 C96ECW 44397809 IC50 = 29.6 nM T22939 CCFG58 44397844 IC50 = 137.3 nM T22939 CTJ6I1 44397845 IC50 = 3000 nM T22939 CL1TE3 44397885 IC50 = 106 nM T22939 CC3XS9 44397913 IC50 = 295.4 nM T22939 C3KL0E 44397914 IC50 = 206.6 nM T22939 C46JYR 44397927 IC50 = 83.6 nM T22939 C0JXT8 44397937 IC50 = 425.6 nM T22939 C04YMW 44397949 IC50 = 24.8 nM T22939 C70AYI 44397969 IC50 = 100 nM T22939 CHJE54 44397984 IC50 = 175.4 nM T22939 CVFX74 44399035 Ki = 39.81 nM T22939 CDR86W 44399036 Ki = 100 nM T22939 CG0U1L 44399066 Ki = 39.81 nM T22939 CY19FD 44399113 Ki = 398.11 nM T22939 C0G6HZ 44399131 Ki = 39.81 nM T22939 C8MDW3 44399211 Ki = 1995.26 nM T22939 C68XGU 44399228 Ki = 100 nM T22939 CXI97U 44402746 IC50 > 1000 nM T22939 CGRX27 44402769 IC50 > 1000 nM T22939 C9XS4E 44402799 IC50 > 1000 nM T22939 CP2IG4 44402961 IC50 = 2000 nM T22939 CXHF58 44403036 IC50 = 36 nM T22939 C25YCZ 44403037 IC50 > 2000 nM T22939 C6JNI4 44403038 IC50 = 85 nM T22939 C45SOW 44403039 IC50 = 210 nM T22939 C2D6VW 44413624 Ki = 39.81 nM T22939 C5DIN3 44413625 Ki = 50.12 nM T22939 C3X4BN 44413631 IC50 = 398.11 nM T22939 CB59JU 44413632 Ki = 63.1 nM T22939 CQI4V7 44413641 Ki = 630.96 nM T22939 CM2XW0 44413744 Ki = 199.53 nM T22939 C9QZ4R 44413757 IC50 = 501.19 nM T22939 CGBV54 44413758 Ki = 316.23 nM T22939 CR7NO0 44413759 Ki = 63.1 nM T22939 C1U0JT 44413770 Ki = 50.12 nM T22939 CH1R7M 44420600 EC50 > 10 nM T22939 CF8N9J 44425531 IC50 = 19 nM T22939 CQ6R5N 44425537 IC50 = 9.6 nM T22939 CGY0M9 44425538 IC50 = 9.3 nM T22939 C6RGU2 44425539 IC50 = 185 nM T22939 CT7LE3 44425540 IC50 > 1000 nM T22939 CT8Q9O 44425541 IC50 = 600 nM T22939 CE53FQ 44425542 IC50 > 1000 nM T22939 C8HO4K 44426782 Ki = 7050 nM T22939 CZM7N0 44430346 IC50 = 1.4 nM T22939 C2AJC1 44430347 IC50 = 1.1 nM T22939 C65HXP 44430353 IC50 = 8.6 nM T22939 C7O2JW 44430354 IC50 = 5.8 nM T22939 CK8QX3 44430355 IC50 = 3.2 nM T22939 CNB12D 44430370 IC50 = 1 nM T22939 CE36SB 44430377 IC50 = 12.5 nM T22939 CTS68I 44430382 IC50 = 2.9 nM T22939 C8BGC1 44430384 IC50 = 2.7 nM T22939 CI8JL5 44430385 IC50 = 0.61 nM T22939 CJ18XT 44430386 IC50 = 0.94 nM T22939 CG8KY9 44430387 IC50 = 1.6 nM T22939 CWR5Z1 44430388 IC50 = 3.2 nM T22939 CBST28 44430389 IC50 = 3.7 nM T22939 CUE9V4 44430390 IC50 = 19.5 nM T22939 C5CB2P 44430391 IC50 = 0.91 nM T22939 CV1DG2 44430392 IC50 = 34 nM T22939 C74CQT 44430393 IC50 = 21 nM T22939 CV6CM4 44430394 IC50 = 39 nM T22939 CEO60C 44430395 IC50 = 1.6 nM T22939 CIOW01 44431179 IC50 > 2000 nM T22939 CR3OW8 44433502 IC50 < 1000 nM T22939 C1Z0QH 44433503 IC50 < 1000 nM T22939 C3SJ5V 44433504 Ki = 313 nM T22939 C3MDG1 44434091 IC50 = 3250 nM T22939 C58WSK 44434092 IC50 = 9460 nM T22939 C0BZA5 44434093 IC50 = 5520 nM T22939 CSA20N 44434095 IC50 > 10000 nM T22939 C2SCP7 44435606 IC50 > 1600 nM T22939 CH5E3L 44435611 IC50 > 1300 nM T22939 CDO62N 44435656 IC50 > 2000 nM T22939 C9TP4C 44435662 IC50 = 1800 nM T22939 C19TMW 44435663 IC50 > 2000 nM T22939 C90WUC 44435667 IC50 = 325 nM T22939 CHFB89 44435668 IC50 = 390 nM T22939 C8IWK2 44435669 IC50 = 1800 nM T22939 CQ6YW8 44436604 EC50 = 2.7 nM T22939 C1XD8O 44436607 EC50 = 49.3 nM T22939 CV3P8M 44436609 EC50 = 62.5 nM T22939 CE64VP 44436611 IC50 = 33.7 nM T22939 C0QN3G 44436614 IC50 = 3.6 nM T22939 CM5TZ0 44436615 IC50 = 10.9 nM T22939 CY3SU6 44436620 IC50 = 11.7 nM T22939 CF71TB 44436622 EC50 = 0.5 nM T22939 CM53RO 44436624 EC50 = 1 nM T22939 CLJF51 44438245 IC50 = 3000 nM T22939 CABV43 44438246 IC50 = 3000 nM T22939 CYK3O2 44438267 IC50 = 71.8 nM T22939 C9PW8F 44438268 IC50 = 1000 nM T22939 C12EVO 44438269 IC50 = 37.1 nM T22939 C8SG5B 44441950 IC50 = 763 nM T22939 CWKU75 44441951 IC50 = 308 nM T22939 C9EG5T 44441952 IC50 = 381 nM T22939 CV0UD9 44441953 IC50 = 141 nM T22939 C1OCJ7 44441954 IC50 = 101 nM T22939 CWH06J 44441955 IC50 = 275 nM T22939 C9IS3X 44441956 IC50 = 9.9 nM T22939 CJQ5G8 44441958 IC50 > 1000 nM T22939 CU32PK 44441961 IC50 = 1.6 nM T22939 CJ5E0V 44441962 IC50 > 1000 nM T22939 CMV0G6 44443285 IC50 = 0.34 nM T22939 CM2JI8 44443286 IC50 = 0.59 nM T22939 CAS57C 44443287 IC50 = 82 nM T22939 CQY8H1 44443288 IC50 = 0.98 nM T22939 C4NQ1C 44443289 IC50 = 0.63 nM T22939 C0WMP8 44443290 IC50 = 18 nM T22939 CQ0N2S 44443291 IC50 = 1 nM T22939 CW30DO 44443292 IC50 = 4.6 nM T22939 CGY14L 44446539 EC50 = 513 nM T22939 C10VES 44446541 EC50 = 10.6 nM T22939 CQ0MN7 44446542 EC50 = 222 nM T22939 CK10ZT 44446543 EC50 = 4450 nM T22939 C2O7ZR 44446546 EC50 = 450 nM T22939 COHW83 44446547 EC50 = 10.3 nM T22939 CBRJ46 44446548 EC50 = 598 nM T22939 C57YRB 44446549 IC50 = 314 nM T22939 CJUK19 44446553 EC50 = 1340 nM T22939 CO6QW4 44446555 EC50 = 54 nM T22939 CH5YR1 44446556 EC50 = 2 nM T22939 CXNA16 44446557 EC50 = 9.8 nM T22939 CX24DP 44446558 EC50 = 198 nM T22939 C5Y2PH 44446559 EC50 = 38 nM T22939 C1WY6L 44446560 EC50 = 1.6 nM T22939 CC0XY9 44446561 EC50 = 993 nM T22939 C6H1FC 44446562 EC50 = 19 nM T22939 CUZ20D 44446563 EC50 > 1000 nM T22939 CA52JZ 44446564 EC50 = 258 nM T22939 CUY6O3 44451244 EC50 = 0.15 nM T22939 CFL39X 44451259 EC50 = 1 nM T22939 CF1IW6 44451277 EC50 = 1.13 nM T22939 C35LBA 44451278 EC50 = 0.29 nM T22939 CRXU40 44451295 EC50 = 2.54 nM T22939 C7B5KA 44451321 EC50 = 0.36 nM T22939 CTC03X 44451341 EC50 = 4 nM T22939 C0NVY8 44451358 EC50 = 2.6 nM T22939 CLT2E4 44451378 EC50 = 0.49 nM T22939 C5D0SE 44451380 EC50 = 1.1 nM T22939 CYK7E9 44451381 EC50 = 0.74 nM T22939 C92GKF 44451394 EC50 = 0.12 nM T22939 CEA31B 44451395 EC50 = 1.3 nM T22939 CE60HQ 44451409 EC50 = 0.23 nM T22939 CX5Y7M 44451461 IC50 = 0.2 nM T22939 C9JT2Q 44451462 IC50 = 0.2 nM T22939 CM52WP 44451463 EC50 = 0.49 nM T22939 CO0KE6 44451464 IC50 = 0.43 nM T22939 C3WH2N 44451475 IC50 = 0.75 nM T22939 CO34KJ 44457134 IC50 = 48 nM T22939 CYG7X4 44473146 IC50 > 10000 nM T22939 CR5SI0 44476535 EC50 > 10000 nM T22939 CM29JD 44516036 IC50 = 8280 nM T22939 C8EHC4 44517745 EC50 = 1.6 nM T22939 CY6F7K 44517750 EC50 = 0.5 nM T22939 CA0S9F 44517751 IC50 = 8 nM T22939 CTRB23 44517777 EC50 = 0.3 nM T22939 C83JWO 44517778 EC50 = 0.3 nM T22939 CR19IH 44543858 IC50 > 2000 nM T22939 C05HEP 44543860 IC50 > 2000 nM T22939 C45ZHO 44543969 IC50 > 2000 nM T22939 C25OXZ 44544094 IC50 > 2000 nM T22939 C7JIF6 44544321 IC50 > 2000 nM T22939 CWP18J 44560815 EC50 = 10.7 nM T22939 CGF03I 44561102 IC50 = 104.7 nM T22939 CF6V4G 44563171 EC50 > 10000 nM T22939 CX34IK 44564027 IC50 = 1.3 nM T22939 CK8MH3 44565647 Ki = 34 nM T22939 CR1EX0 44568002 IC50 = 10000 nM T22939 C9KPI1 44568003 IC50 = 6800 nM T22939 C3ZP4C 44568040 IC50 = 3400 nM T22939 C4H8BI 44568041 IC50 = 1600 nM T22939 CSNV65 44568081 IC50 = 250 nM T22939 C6D9GJ 44568082 IC50 = 1000 nM T22939 CP19AM 44568083 IC50 = 400 nM T22939 CHM92V 44568084 IC50 = 2100 nM T22939 CR9NZ7 44568085 IC50 = 1100 nM T22939 C72SHF 44568120 IC50 = 120 nM T22939 C0SYE1 44568121 IC50 = 150 nM T22939 CB7I3F 44568122 IC50 = 690 nM T22939 C2LB4X 44568123 IC50 = 450 nM T22939 CG79ZB 44579751 EC50 = 3.3 nM T22939 CT0FD9 44579819 IC50 = 14.3 nM T22939 CG83KV 44579820 IC50 = 197.4 nM T22939 CT8C4J 44579838 IC50 = 175.1 nM T22939 CV75OH 44579839 IC50 = 500 nM T22939 CZPM61 44579855 IC50 = 17.1 nM T22939 C6BZW1 44579856 IC50 = 10 nM T22939 CXD4E0 44585534 IC50 = 207.7 nM T22939 CR0JY4 44585535 IC50 = 65.2 nM T22939 C7NG5L 44585536 IC50 = 88 nM T22939 CNHJ31 44585548 IC50 = 100 nM T22939 C9QDJ2 44585549 IC50 = 1000 nM T22939 CI9KT2 44585550 IC50 = 1000 nM T22939 CRT56J 44585551 IC50 = 29.9 nM T22939 CJ7T5O 44585552 IC50 = 107.6 nM T22939 C8BGL6 44585565 IC50 = 13.3 nM T22939 CY6CF7 44585566 IC50 = 22.5 nM T22939 C45TDP 44585567 IC50 = 82.4 nM T22939 C9G5OI 44585568 IC50 = 34.1 nM T22939 CS81IL 44587000 IC50 = 394 nM T22939 C71CKD 44587057 IC50 > 1000 nM T22939 C2USW6 44587219 IC50 > 1000 nM T22939 CUA45E 44587248 IC50 = 120 nM T22939 C91YAW 44587251 IC50 = 176 nM T22939 CJ3VI8 44593465 Ki = 35 nM T22939 CIJP09 44605898 EC50 = 0.3 nM T22939 CT5G6Z 45101436 EC50 = 0.7943 nM T22939 C9PLK4 45263610 IC50 = 620 nM T22939 C78JKD 45265930 IC50 = 170 nM T22939 C51HCA 45267201 EC50 = 6 nM T22939 C26QAU 45267222 EC50 = 6.8 nM T22939 C65IKR 45267223 IC50 = 200 nM T22939 C8UN2F 45267226 IC50 = 398 nM T22939 C1Z9XI 45267345 IC50 = 930 nM T22939 CWKP29 45267349 IC50 = 0.3 nM T22939 CN8HI2 45267356 IC50 > 1000 nM T22939 CG6X9E 45267360 IC50 > 1000 nM T22939 C2B0JK 45267748 IC50 = 3000 nM T22939 CW15SE 45267757 IC50 = 25 nM T22939 C1TVR0 45267765 IC50 = 63 nM T22939 CMF7N4 45268071 IC50 = 50 nM T22939 C9K7GN 45268072 EC50 = 1.3 nM T22939 CPQF40 45268078 IC50 = 32 nM T22939 CV4AN2 45268083 EC50 = 0.05 nM T22939 C1A4TO 45268599 IC50 = 200 nM T22939 C3WV4T 45268600 EC50 = 625 nM T22939 CE83JD 45268636 IC50 = 400 nM T22939 C14UWH 45268950 EC50 = 0.6 nM T22939 CF3XL2 45268951 EC50 = 14 nM T22939 CD7T3W 45269091 IC50 = 33 nM T22939 C97ZET 45269449 EC50 = 30 nM T22939 CZ75WU 45269455 EC50 = 70 nM T22939 C87JQL 45269462 EC50 = 0.8 nM T22939 CEF1W0 45269477 IC50 = 250 nM T22939 CCKE74 45269799 EC50 = 272 nM T22939 CMG2Z9 45269807 EC50 = 9.5 nM T22939 C21HYG 45269951 IC50 = 56 nM T22939 CAP56V 45269952 IC50 > 1000 nM T22939 CKG49L 45269958 IC50 = 280 nM T22939 COV60G 45270312 IC50 = 79 nM T22939 CX7JY3 45270332 IC50 = 20 nM T22939 CCER05 45270638 IC50 = 500 nM T22939 CIR20D 45270774 IC50 = 36 nM T22939 C9D1IT 45270779 IC50 = 3.3 nM T22939 CT4I0U 45271113 EC50 = 0.3 nM T22939 CU61RS 45271119 IC50 = 25 nM T22939 C9RFM3 45271120 EC50 = 1415 nM T22939 C4XQD0 45271124 EC50 = 750 nM T22939 CK68ZG 45271140 IC50 = 40 nM T22939 C4TS9W 45271144 IC50 = 400 nM T22939 CPM4S2 45271152 EC50 = 200 nM T22939 CBK7C9 45271451 EC50 = 0.6 nM T22939 C7ZI3A 45271452 IC50 = 25 nM T22939 CCG8U7 45271461 EC50 = 157 nM T22939 CZ2V7P 45271462 EC50 = 3 nM T22939 CJKN81 45271616 IC50 = 7 nM T22939 CF7IB2 45272011 EC50 = 0.8 nM T22939 CEZY97 45272012 EC50 = 2 nM T22939 C08UBE 45272032 IC50 = 125 nM T22939 CEV17D 45272033 IC50 = 1300 nM T22939 CSUI94 45272049 IC50 = 160 nM T22939 CFOM86 45272341 EC50 = 0.7 nM T22939 CAV9J5 45272342 IC50 = 13 nM T22939 CW0TC6 45272345 EC50 = 606 nM T22939 C9P8ZM 45272353 EC50 = 11 nM T22939 C25KCQ 45272356 EC50 = 4.7 nM T22939 C2A9PV 45272364 IC50 = 398 nM T22939 C9MF3P 45272514 IC50 = 82 nM T22939 CT5KW9 45272826 EC50 = 135 nM T22939 C4IFO2 45272879 IC50 = 13 nM T22939 C3DV7O 45273222 EC50 = 0.02 nM T22939 CZP8X3 45273223 EC50 = 0.04 nM T22939 C5JXA2 45273230 EC50 = 0.02 nM T22939 CUZ5C6 45273374 IC50 = 60 nM T22939 CM1BJ8 45273809 IC50 = 40 nM T22939 CTD93Q 45273810 IC50 = 50 nM T22939 C57EZH 45275745 IC50 = 9800 nM T22939 CN6B0C 45369230 IC50 = 810 nM T22939 CFDP96 45375982 EC50 = 1 nM T22939 C1SPF6 45375983 EC50 = 2 nM T22939 CWG08H 45375985 IC50 = 18 nM T22939 C1C4ZM 45375986 IC50 = 10 nM T22939 C4Y5DE 45483811 IC50 = 195 nM T22939 CLP82D 45483812 IC50 = 66 nM T22939 C7SL4F 45483819 IC50 = 79 nM T22939 CI97US 45483863 IC50 = 3 nM T22939 C98WDQ 45485494 IC50 = 794.33 nM T22939 CB2LO0 45485501 IC50 = 1000 nM T22939 C96THD 45485556 IC50 = 794.33 nM T22939 CRP29T 45485557 EC50 > 10000 nM T22939 C0WQ4R 45486436 Ki = 451 nM T22939 COG73H 45486437 Ki = 238 nM T22939 C2NWO7 45486438 Ki = 132 nM T22939 CW7J5K 45486451 Ki = 409 nM T22939 CU3IY5 45486473 Ki = 230 nM T22939 CHRX37 45486474 Ki = 1810 nM T22939 CNT32O 46224623 IC50 = 63 nM T22939 CFS6Q5 46224644 EC50 = 11 nM T22939 CURS28 46224649 IC50 = 40 nM T22939 C75QAG 46224653 IC50 = 80 nM T22939 CB5HP0 46224657 EC50 = 3160 nM T22939 CI3OC4 46224664 EC50 = 10 nM T22939 CS9D6X 46224668 IC50 = 12 nM T22939 C5N2WP 46224669 EC50 = 2.1 nM T22939 C6XQF5 46224670 EC50 = 24 nM T22939 C72ZGS 46224672 EC50 = 843 nM T22939 CNG16S 46224673 EC50 = 3 nM T22939 CQ75YZ 46224676 IC50 = 100 nM T22939 CS0Y7O 46224677 EC50 = 364 nM T22939 CJP6A9 46224678 IC50 = 25 nM T22939 CR9J1L 46224680 EC50 = 4 nM T22939 CZS7L4 46224681 EC50 = 3 nM T22939 CJZL72 46224683 EC50 = 1130 nM T22939 CKQF01 46224685 IC50 = 50 nM T22939 C15RNW 46224687 IC50 = 25 nM T22939 C81YIZ 46224688 IC50 = 25 nM T22939 CRSM47 46224691 IC50 = 63 nM T22939 C0RJG8 46224692 EC50 = 0.1 nM T22939 CQC6J0 46224693 IC50 = 50 nM T22939 C2A5QX 46224699 EC50 = 41 nM T22939 CPHQ30 46224702 IC50 = 30 nM T22939 C7JXG3 46224705 EC50 = 8 nM T22939 CMYU19 46224706 EC50 = 0.4 nM T22939 CBNI02 46830477 IC50 = 4820 nM T22939 C1RJV2 46830478 IC50 > 10000 nM T22939 C1BYW8 46830503 IC50 > 10000 nM T22939 C04BWG 46830504 IC50 = 2511.89 nM T22939 CY2ZJ0 46830505 IC50 = 1584.89 nM T22939 CC45TP 46830506 IC50 > 10000 nM T22939 CN7Q8A 46830507 IC50 > 10000 nM T22939 C0QT3G 46830795 IC50 > 10000 nM T22939 C0JCX3 46830796 IC50 = 1995.26 nM T22939 CMS6R9 46830797 IC50 = 6309.57 nM T22939 CJIN74 46830798 IC50 > 10000 nM T22939 CRY31M 46830799 IC50 > 10000 nM T22939 CKA07I 46830800 IC50 > 10000 nM T22939 C4XRF9 46830801 IC50 > 10000 nM T22939 C2NC3V 46831087 IC50 > 10000 nM T22939 CXP6K3 46831397 IC50 = 2511.89 nM T22939 C0QNC9 46831400 IC50 = 3162.28 nM T22939 CX6L7Q 46831696 IC50 = 1584.89 nM T22939 CQ1IP3 46831697 IC50 = 5011.87 nM T22939 CL1KR4 46831698 IC50 = 794.33 nM T22939 C1DH9W 46831699 IC50 = 630.96 nM T22939 CASV14 46831700 IC50 > 10000 nM T22939 CTXY26 46831701 IC50 > 10000 nM T22939 CG0J5K 46831956 IC50 > 10000 nM T22939 CY3WK4 46831957 IC50 > 10000 nM T22939 CP19UN 46831958 IC50 > 10000 nM T22939 CBJZ85 46831959 IC50 > 2511.89 nM T22939 CE4VC8 46831960 IC50 > 10000 nM T22939 CAR23U 46832233 IC50 > 10000 nM T22939 CUAO43 46832234 IC50 > 10000 nM T22939 CM40EP 46832235 IC50 > 2511.89 nM T22939 CJ32XT 46832236 IC50 > 10000 nM T22939 C81GUN 46832237 IC50 > 10000 nM T22939 CT31AL 46832511 IC50 = 794.33 nM T22939 CR15XE 46832512 IC50 > 10000 nM T22939 CW12GM 46832513 IC50 > 10000 nM T22939 C0GTK8 46832514 IC50 > 10000 nM T22939 C8HO0L 46832515 IC50 > 10000 nM T22939 C2S6PL 46834818 IC50 = 4400 nM T22939 C9ZWM8 46866594 IC50 = 1200 nM T22939 CD04CW 46871871 Ki = 35 nM T22939 CXD42C 46871872 Ki = 84 nM T22939 C7KW8T 46883839 EC50 > 19952.62 nM T22939 CZSG25 46883893 EC50 > 10000 nM T22939 CMR49F 46885348 IC50 = 10000 nM T22939 C4TLX3 46885390 IC50 = 7900 nM T22939 CSP3D8 46885467 IC50 = 7800 nM T22939 CP3O2L 46885469 IC50 = 8600 nM T22939 CG6JE7 46885508 IC50 = 8300 nM T22939 CX2U0L 46886033 IC50 = 1400 nM T22939 C6J5RT 46886034 IC50 = 2500 nM T22939 C72MUY 46889765 IC50 = 131 nM T22939 CV3BA5 46889766 IC50 = 13 nM T22939 C79OZG 46889803 IC50 > 10000 nM T22939 CD28AJ 46889804 IC50 = 173 nM T22939 CV53NK 46889805 IC50 = 35 nM T22939 C8FTP4 46889806 IC50 = 886 nM T22939 CY37VP 46889807 IC50 = 56 nM T22939 CH48WI 46889808 IC50 = 1130 nM T22939 CJC1W6 46889847 IC50 = 204 nM T22939 C6DVO1 46889848 IC50 = 47 nM T22939 CPH7G8 46889849 IC50 = 71 nM T22939 CZ90FC 46894119 IC50 > 25000 nM T22939 CJW14R 46905371 Ki = 0.4 nM T22939 C8T6RN 46906110 Ki = 78 nM T22939 CP04YQ 46906111 Ki = 58 nM T22939 C4RFX9 46906112 Ki = 87 nM T22939 CCM4H0 46906113 Ki = 47 nM T22939 C32JOS 46906137 Ki = 85 nM T22939 C3GP8J 46906138 Ki = 56 nM T22939 CT0QU8 46906139 Ki = 31 nM T22939 C16CJP 46906140 Ki = 18 nM T22939 CM4H3Y 46906173 Ki = 80 nM T22939 CU9H2X 46906174 Ki = 66 nM T22939 CQ2PU6 46906175 Ki = 13 nM T22939 C42RPK 46906176 Ki = 10.8 nM T22939 CZ7OE3 46906177 Ki = 10.2 nM T22939 CAK8Y1 46906229 Ki = 8.5 nM T22939 CE1DN6 46906230 Ki = 11.2 nM T22939 CT57UI 46906231 Ki = 9.1 nM T22939 C09VDP 46906256 Ki = 13 nM T22939 CAQT54 46906257 Ki = 28 nM T22939 CV84RA 46906258 Ki = 51 nM T22939 CKTU08 46906259 Ki = 99 nM T22939 CGW15V 46906285 Ki > 10000 nM T22939 COMC86 46906286 Ki = 444 nM T22939 CF0UH7 46906482 Ki = 103 nM T22939 C3RVF1 46906483 Ki = 75 nM T22939 CID4F9 46906484 Ki = 1119 nM T22939 CSK01Q 46906501 Ki = 173 nM T22939 C7ELM3 46906502 Ki = 121 nM T22939 CRH1T2 46906503 Ki = 35 nM T22939 C81MYC 46906504 Ki = 46 nM T22939 CAS06I 46906529 Ki = 36 nM T22939 C0I5SR 46906530 Ki = 49 nM T22939 C7BVX3 46906531 Ki = 68 nM T22939 C4BM6J 46906561 Ki = 43 nM T22939 CEP63J 46906562 Ki = 50 nM T22939 CJ9EN0 46906563 Ki = 76 nM T22939 C3Q7RI 46913890 IC50 = 2010 nM T22939 CP91XE 46914741 IC50 = 3180 nM T22939 CTM2J5 46915203 IC50 = 2080 nM T22939 C75IFZ 46915353 IC50 > 4310 nM T22939 CX70GY 46915355 IC50 = 1030 nM T22939 C7NC4B 46917090 IC50 = 2480 nM T22939 C2LCJ7 46937290 IC50 = 1200 nM T22939 CKQ8J3 46937431 IC50 > 2000 nM T22939 CL7P3N 46938234 IC50 = 2529 nM T22939 COS28G 46938235 IC50 = 6810 nM T22939 CFJT93 46938236 IC50 = 1590 nM T22939 CHL70M 46938239 IC50 = 831 nM T22939 C8P7JH 46938914 IC50 > 2000 nM T22939 CY95VK 46938915 IC50 > 2000 nM T22939 CVX25Q 46938916 IC50 = 1900 nM T22939 C2V5AT 46939019 IC50 = 1200 nM T22939 C5R6GI 46939020 IC50 > 2000 nM T22939 CF1BX0 46939115 IC50 > 2000 nM T22939 C4P0EU 46939116 IC50 = 1300 nM T22939 CD6B7X 46939395 IC50 = 600 nM T22939 C1KXF2 46939396 IC50 > 2000 nM T22939 CU3S6H 49836028 Ki = 53 nM T22939 C96SLW 49851364 Ki = 273 nM T22939 CDN4K6 49851369 Ki = 31 nM T22939 C0K7OD 49851464 Ki = 144 nM T22939 C4YXN1 49851467 Ki = 55 nM T22939 CI0MX2 49851469 Ki = 140 nM T22939 CUD91T 49862248 EC50 > 10000 nM T22939 CCH43Y 49862353 IC50 = 36 nM T22939 CSK80N 49862354 IC50 = 27 nM T22939 CN6VJ1 49862355 IC50 = 24 nM T22939 C7CT5G 49862415 IC50 = 47 nM T22939 C90TAD 49862416 IC50 = 118 nM T22939 CTKV39 49864176 IC50 = 1880 nM T22939 CZ8J1V 50942115 Ki = 1200 nM T22939 C23OEF 50942312 EC50 > 10000 nM T22939 CGKT15 51003433 IC50 = 3060 nM T22939 CX1KO8 51346768 Ki = 0.214 nM T22939 C7N9TD 51346823 Ki = 2095 nM T22939 C0WDX3 51347001 Ki = 231 nM T22939 CF8DK7 51347002 Ki = 680 nM T22939 CTH45Q 52918523 IC50 > 10000 nM T22939 CEC4I7 52941608 IC50 > 2000 nM T22939 CDV90J 52942528 IC50 > 1000 nM T22939 C8Y9SU 52944898 IC50 > 1000 nM T22939 CTV7K1 53316621 EC50 = 199.53 nM T22939 CLC5U1 53316851 EC50 = 251.19 nM T22939 C82ATJ 53316852 EC50 = 794.33 nM T22939 CK5UT4 53317489 Ki = 0.298 nM T22939 C9Y0RM 53318166 EC50 = 630.96 nM T22939 CCT76B 53318167 EC50 > 10000 nM T22939 CQI41V 53318658 Ki = 3000 nM T22939 CM0LU1 53318659 Ki = 1100 nM T22939 CVIE23 53319666 Ki = 190 nM T22939 CUD48O 53320087 Ki = 454 nM T22939 C7VWT1 53322135 EC50 = 199.53 nM T22939 C8MU3A 53322265 IC50 = 3220 nM T22939 CJD29K 53323475 EC50 = 7.943 nM T22939 CD0N1K 53323476 EC50 > 10000 nM T22939 C16TGD 53325224 Ki = 1900 nM T22939 CIU8H2 53325583 EC50 = 125.89 nM T22939 CLG69E 53325612 EC50 = 50.12 nM T22939 CYH3V0 53325642 Ki = 478 nM T22939 CP7Y9M 53326069 EC50 = 79.43 nM T22939 C82DYI 53326614 Ki = 28 nM T22939 CJCP75 53359074 Ki = 1829 nM T22939 C01IUW 53379592 IC50 = 1280 nM T22939 CVX25U 53379593 IC50 = 140 nM T22939 CSF57P 53379700 IC50 = 10000 nM T22939 C39UJI 53379701 IC50 = 50500 nM T22939 CUR24K 53875787 IC50 = 130 nM T22939 C2P5HX 54582225 IC50 = 410 nM T22939 CQ02IF 54582227 IC50 = 560 nM T22939 CS9O7F 54582228 IC50 = 5800 nM T22939 CX6S5F 54584172 IC50 = 1100 nM T22939 CGOZ54 54585120 IC50 = 4000 nM T22939 C8P9ZJ 54586082 IC50 = 12000 nM T22939 CPF9X2 54587076 IC50 = 2700 nM T22939 C30XLO 54592009 IC50 > 10000 nM T22939 CX4V9H 56589542 IC50 = 123 nM T22939 CCJ42Y 56589543 IC50 = 500 nM T22939 CT2B1S 56593207 IC50 = 220 nM T22939 C9W5DZ 56593984 Ki = 1228 nM T22939 CA9ER8 56594118 Ki = 1829 nM T22939 CI0FV7 56594209 IC50 = 500 nM T22939 CB4M7S 56594210 IC50 = 860 nM T22939 C0AF7Z 56594211 IC50 = 510 nM T22939 C1MAK4 56594212 IC50 = 470 nM T22939 C1MZS2 56594213 IC50 = 390 nM T22939 CC6ML8 56594214 IC50 = 400 nM T22939 CCJ9A8 56594215 IC50 = 770 nM T22939 CA81TE 56594346 IC50 = 630 nM T22939 C47KYA 56594347 IC50 = 380 nM T22939 CG5DE6 56594348 IC50 = 360 nM T22939 C5V1ES 56594349 IC50 = 250 nM T22939 CX4AD2 56594350 IC50 = 470 nM T22939 CDSF79 56594351 IC50 = 260 nM T22939 CM30AD 56594352 IC50 = 880 nM T22939 CX2A1U 56594353 IC50 = 1280 nM T22939 C3NS2R 56594474 IC50 = 3340 nM T22939 CQB1N0 56594475 IC50 = 2590 nM T22939 CHM1C9 56594476 IC50 = 290 nM T22939 CZIE68 56594477 IC50 = 310 nM T22939 CY5T0V 56594478 IC50 = 210 nM T22939 CR9AL1 56594479 IC50 = 1110 nM T22939 CCS5A6 56594480 IC50 = 560 nM T22939 CV90SA 56594481 IC50 = 190 nM T22939 CR4U9K 56594613 IC50 = 220 nM T22939 C02FMR 56661892 IC50 = 27900 nM T22939 CF3G2M 56925477 IC50 = 350 nM T22939 CZ7O8G 56925478 IC50 = 1400 nM T22939 CW87RG 56925573 IC50 = 1600 nM T22939 C30DAL 56925669 IC50 > 10000 nM T22939 CQHA65 56925670 IC50 > 10000 nM T22939 CJP31U 56925671 IC50 > 10000 nM T22939 CI3S6F 56925790 IC50 > 10000 nM T22939 CTY1Q9 56925791 IC50 > 10000 nM T22939 CTG9I7 56926011 IC50 = 930 nM T22939 CY3B1Z 57330204 IC50 = 2300 nM T22939 CX6Q9M 57390301 Ki = 310 nM T22939 C3Y9SF 57390753 IC50 = 85 nM T22939 C7R4HE 57390754 IC50 = 41 nM T22939 CM0SG2 57390990 IC50 = 1200 nM T22939 CNTL28 57392477 IC50 = 771 nM T22939 C4SD8X 57392560 IC50 = 65 nM T22939 CU8AN3 57392780 IC50 = 1000 nM T22939 CX12JM 57392781 IC50 = 155 nM T22939 C9OMW1 57392782 IC50 = 1400 nM T22939 CP26TS 57394182 IC50 = 307 nM T22939 C8S0HJ 57394288 IC50 = 35 nM T22939 C30JOV 57394501 IC50 = 207 nM T22939 CINU04 57396254 IC50 = 440 nM T22939 C1O6JU 57396255 IC50 = 745 nM T22939 C24YLG 57399054 Ki = 285 nM T22939 COU74V 57399417 IC50 = 430 nM T22939 C54BJR 57399499 IC50 = 46 nM T22939 CVOB64 57399718 IC50 > 2000 nM T22939 CF83VM 57401459 Ki = 1529 nM T22939 C7W3YD 57401479 IC50 > 2000 nM T22939 C6RX7O 57403004 IC50 = 101 nM T22939 CR6L7E 57403222 IC50 > 2000 nM T22939 CG2J6D 57403536 IC50 = 1372 nM T22939 CPU6W7 57473898 IC50 = 3500 nM T22939 CEJ25K 57473899 IC50 > 2000 nM T22939 CUJ08D 57474008 IC50 = 540 nM T22939 C3WG0L 57666312 Ki = 970 nM T22939 C43GDR 57666397 Ki = 750 nM T22939 CTM6K5 57690900 IC50 = 4500 nM T22939 C1KZT3 57906156 IC50 > 10000 nM T22939 C3IN9F 57983276 IC50 > 10000 nM T22939 CJ6Y1B 58026134 IC50 > 2000 nM T22939 CV1RX3 58026153 IC50 > 2000 nM T22939 C19XQV 58026164 IC50 > 2000 nM T22939 CR7H3O 58026170 IC50 > 2000 nM T22939 C7XL3D 58026176 IC50 > 2000 nM T22939 CT1EM3 58064710 IC50 = 1490 nM T22939 C8S3EQ 58064714 IC50 = 494 nM T22939 CPI62D 58064720 IC50 = 684 nM T22939 CL42XF 58064726 IC50 = 597 nM T22939 CPL9A6 58064729 IC50 = 806 nM T22939 CRFS78 58064730 IC50 = 550 nM T22939 CN1J3V 58064734 IC50 = 3670 nM T22939 CA0SH5 58064735 IC50 = 2600 nM T22939 CI7BP4 58064741 IC50 = 5310 nM T22939 C2FZA7 58064756 IC50 = 1520 nM T22939 C4C2FT 58599563 IC50 = 1400 nM T22939 CI6XF5 58742295 IC50 = 321 nM T22939 C0JL7A 58973277 IC50 > 1000 nM T22939 CN3YR2 59233334 Ki = 1194 nM T22939 CY38HG 59233337 Ki > 1250 nM T22939 CUX4E7 59233347 Ki > 1250 nM T22939 CO63VJ 59233364 Ki > 1250 nM T22939 C2A9JO 59251119 Ki > 5000 nM T22939 CD8A6P 59281281 IC50 = 390 nM T22939 CBZ0M5 59281312 IC50 > 10000 nM T22939 CCT59B 59281329 IC50 = 5600 nM T22939 CQI5C4 59281343 IC50 = 1300 nM T22939 CPE83R 59281354 IC50 = 1600 nM T22939 CI9EP1 59281363 IC50 = 1100 nM T22939 CQ2BO1 59281403 IC50 = 2400 nM T22939 CP78RD 59281411 IC50 = 2500 nM T22939 CCNU12 59281412 IC50 = 370 nM T22939 C7HVB1 59281416 IC50 = 4600 nM T22939 CE5A0V 59281447 IC50 = 5400 nM T22939 CZT9S6 59281449 IC50 > 10000 nM T22939 CIKQ89 59281508 IC50 > 10000 nM T22939 CE1A7J 59281531 IC50 > 10000 nM T22939 CK9JZ4 59281538 IC50 = 1700 nM T22939 C4TG5U 59281540 IC50 = 4000 nM T22939 CPC80S 59281541 IC50 = 2000 nM T22939 CXS5C4 59281543 IC50 > 10000 nM T22939 C7KPR9 59281566 IC50 = 2500 nM T22939 CUJP64 59281599 IC50 = 2300 nM T22939 CYZI85 59556974 EC50 > 10000 nM T22939 C5C3AO 59770003 Ki = 99 nM T22939 C2TNO8 60026286 IC50 > 2000 nM T22939 CZE5J8 60026377 IC50 > 2000 nM T22939 CJ34GW 60026481 IC50 = 1100 nM T22939 CJ7E6C 60026483 IC50 > 2000 nM T22939 C0LDS2 60026592 IC50 > 2000 nM T22939 C31PTC 60026641 IC50 > 2000 nM T22939 C67NSE 60026675 IC50 > 2000 nM T22939 C6GP5R 60026731 IC50 = 780 nM T22939 C5M8HV 60026772 IC50 = 880 nM T22939 CI36XS 60026787 IC50 > 2000 nM T22939 C3JD8M 60026802 IC50 > 2000 nM T22939 CE9MI4 60026817 IC50 > 2000 nM T22939 C3UQ8M 60026849 IC50 = 1000 nM T22939 C04EKW 60026878 IC50 > 2000 nM T22939 CM3Y0X 60026895 IC50 > 2000 nM T22939 C1L4JR 60165333 IC50 = 5000 nM T22939 C1CXY9 66996546 IC50 > 10000 nM T22939 CH39DP 67053383 IC50 > 2000 nM T22939 C3LF8O 67053425 IC50 > 2000 nM T22939 CNQ8T5 69571559 IC50 > 2000 nM T22939 CARO49 70685018 Ki = 0.48 nM T22939 C5QPC0 70697572 Ki = 1.7 nM T22939 CUH71V 71239417 IC50 = 700 nM T22939 C94FCP 71452686 IC50 = 130 nM T22939 CF08ME 71457470 Ki = 478 nM T22939 CEO5G4 71461616 IC50 = 65 nM T22939 C1MHC0 71467246 IC50 = 5400 nM T22939 C4B0IC 71467248 IC50 = 4200 nM T22939 CYW34A 71519686 IC50 = 3200 nM T22939 CGK4S8 71543393 Ki = 872 nM T22939 C83YJF 71544946 IC50 > 5000 nM T22939 CT9Y5D 71549558 IC50 = 2400 nM T22939 C8ZX0F 71549573 IC50 = 3600 nM T22939 CZ8Y7O 71549829 IC50 = 1900 nM T22939 CPFL57 71549843 IC50 = 8100 nM T22939 CY8SP0 71549969 IC50 = 8200 nM T22939 CX6JR5 71550242 IC50 = 2900 nM T22939 C6WIA2 71550244 IC50 = 2900 nM T22939 CSHT69 71550657 IC50 > 5000 nM T22939 C1JP3D 71712294 Ki = 312.5 nM T22939 CP5KM8 72163477 IC50 = 4600 nM T22939 CA6O4K 72163478 IC50 = 1800 nM T22939 C27XWS 72163479 IC50 = 1000 nM T22939 C6M9CN 72163480 IC50 = 740 nM T22939 CL8AH4 72163481 IC50 = 5000 nM T22939 CB2SD9 72163621 IC50 = 2200 nM T22939 CU6NA8 72163622 IC50 = 61 nM T22939 CTEV75 72163623 IC50 = 770 nM T22939 CER73F 72163624 IC50 = 400 nM T22939 CC8VM7 72163625 IC50 > 10000 nM T22939 CS69AC 72163626 IC50 = 5600 nM T22939 CAJ0H5 72163627 IC50 = 4900 nM T22939 C1D3EU 72163754 IC50 = 3200 nM T22939 C1G3ES 72163755 IC50 = 1600 nM T22939 CP8AC2 72188914 Ki = 107 nM T22939 CA6FO5 72188915 Ki = 56 nM T22939 C34FBN 72544603 IC50 > 9211 nM T22939 CLA3Y9 72710581 Ki = 26.8 nM T22939 CXB45U 72724690 IC50 = 620 nM T22939 CI2K6C 72725442 IC50 = 4200 nM T22939 C0W2UD 72725443 IC50 = 5500 nM T22939 CQ5D1B 72725444 IC50 = 3400 nM T22939 C2PJV7 72725445 IC50 > 10000 nM T22939 CQ4Z2C 72725446 IC50 = 2000 nM T22939 C47IMQ 72725447 IC50 = 8200 nM T22939 CJSK52 72725491 IC50 = 7400 nM T22939 CS6J4T 72725492 IC50 = 3400 nM T22939 C41FYD 72725493 IC50 = 1200 nM T22939 CUG96L 72725494 IC50 = 1500 nM T22939 CFHJ16 72725495 IC50 = 720 nM T22939 CW7IY3 72725496 IC50 = 2100 nM T22939 CSV1I7 72725497 IC50 = 860 nM T22939 COV09R 72725548 IC50 > 10000 nM T22939 CTE01I 72725549 IC50 > 10000 nM T22939 C09ZFS 72725550 IC50 = 3500 nM T22939 C2Z7QT 72725551 IC50 = 210 nM T22939 C0K2CP 72725552 IC50 = 6400 nM T22939 C37MEN 72725553 IC50 = 2800 nM T22939 CYSM01 72725554 IC50 = 2500 nM T22939 C3POU0 72736045 Ki = 22 nM T22939 COU49R 76314656 IC50 = 1400 nM T22939 C95NBT 76314657 IC50 > 2000 nM T22939 CZ08OF 76317198 IC50 > 2000 nM T22939 CR5B2V 76317199 IC50 = 5300 nM T22939 C5YFZ6 76318225 IC50 > 2000 nM T22939 C0RK5D 76321918 IC50 > 2000 nM T22939 C3IC5B 76329113 IC50 > 2000 nM T22939 C1RB6X 76329114 IC50 > 2000 nM T22939 CP8M1Z 76332766 IC50 > 2000 nM T22939 CKDI18 76332767 IC50 > 2000 nM T22939 CK21EY 77461202 IC50 = 290 nM T22939 CSP8F2 84482101 IC50 = 510 nM T22939 CIU65X 86280440 Ki = 64.2 nM T22939 CNEP10 86345430 IC50 = 3.467 nM T22939 CT50AL 87539277 IC50 > 1000 nM T22939 CY05IC 87733533 IC50 = 199.53 nM T22939 C9EH7I 89500376 Ki = 1220 nM T22939 C0EQS7 89501406 Ki = 520 nM T22939 C8JG7O 89510193 Ki = 448 nM T22939 CK5D1A 90395281 IC50 = 4900 nM T22939 CQ06RH 90654508 IC50 > 2000 nM T22939 C5E6UV 90656124 IC50 = 3800 nM T22939 C6VZ7X 90656360 IC50 = 2720 nM T22939 CNCB43 90656361 IC50 = 2190 nM T22939 CS42NY 90656362 IC50 = 2040 nM T22939 C6C2ON 100464098 IC50 = 960 nM T22939 CUYX25 100491087 IC50 = 990 nM T22939 CE4Z3U 102313488 IC50 = 240 nM T22939 CT01WS 113098759 IC50 = 62 nM T22939 CFQK93 113098760 IC50 = 740 nM T22939 CF67IH 117917065 Ki = 268 nM T22939 CFG2T8 117917077 Ki = 12380 nM T22939 CDZ31K 117917098 Ki = 282.2 nM T22939 CW27MY 118063735 EC50 > 30000 nM T22939 C9L5EW 118599756 Ki > 50118.72 nM T22939 CREN83 118707969 Ki = 12380 nM T22939 CC2I1P 118707970 Ki = 5043 nM T22939 C7XD9E 118707971 Ki = 2040 nM T22939 CF60IG 118707972 Ki = 5337 nM T22939 CZB1G7 118707973 Ki = 10630 nM T22939 C3XOR9 118707974 Ki = 1168 nM T22939 CDA17Q 118707975 Ki = 2909 nM T22939 CTKA86 118707976 Ki = 5337 nM T22939 CVW2B3 118707977 Ki = 623 nM T22939 CLS7C1 118707978 Ki = 52.8 nM T22939 C9LV0M 118707979 Ki = 44.9 nM T22939 CV4DC0 118707980 Ki = 604.1 nM T22939 COJB29 118707981 Ki = 2322 nM T22939 C3TLR1 118707982 Ki = 33330 nM T22939 CMW3N5 118707983 Ki = 1362 nM T22939 C72VHF 118707984 Ki = 22.7 nM T22939 C06ZWX 118707985 Ki = 106.2 nM T22939 CC2H4E 118714881 IC50 > 10000 nM T22939 C6Y5JG 118723171 IC50 = 1700 nM T22939 CE3I9T 118723172 IC50 > 2000 nM T22939 C13AIC 118723173 IC50 > 2000 nM T22939 C21SWI 118723174 IC50 > 2000 nM T22939 CKR24J 118723175 IC50 > 2000 nM T22939 C28YZF 118723176 IC50 > 2000 nM T22939 C6AGI7 118723177 IC50 > 2000 nM T22939 C4QO8E 118723178 IC50 > 2000 nM T22939 C8ICV0 118727000 IC50 = 53 nM T22939 CA8ZW3 118727001 IC50 = 177.7 nM T22939 CESR95 118727002 IC50 = 58.4 nM T22939 C2DQ8U 118727003 IC50 = 25.8 nM T22939 CZ4V8L 118727004 IC50 = 39.5 nM T22939 C5P0AX 118727005 IC50 = 174.2 nM T22939 CMV85B 118727006 IC50 = 124.6 nM T22939 C7Q4KT 118727007 IC50 = 403.9 nM T22939 C0XKT7 118727008 IC50 = 228 nM T22939 C1S4YN 118727009 IC50 = 25 nM T22939 CN6M9B 118727010 IC50 = 36.2 nM T22939 CVQW86 118727011 IC50 = 118.9 nM T22939 CGD6K3 118727012 IC50 = 74 nM T22939 CU5WB1 118727013 IC50 > 1000 nM T22939 C03GVR 121238090 IC50 = 175 nM T22939 C6TBD2 121345502 EC50 > 20000 nM T22939 C27NGB 121493947 IC50 = 43 nM T22939 CG13LX 122178361 IC50 = 2800 nM T22939 C9LIR4 122179356 Ki = 22 nM T22939 CUI57B 122179357 Ki = 403 nM T22939 CR98CI 122179360 Ki > 1250 nM T22939 CY18QG 122186737 Ki = 4190 nM T22939 C0OR2H 122186738 Ki = 688 nM T22939 CU0Y8B 122186739 Ki = 3940 nM T22939 CWF0Q4 122186740 Ki = 22.3 nM T22939 CBE6Q8 122186741 Ki = 253 nM T22939 CX13DR 122186742 Ki = 4000 nM T22939 CJ74HX 122186743 Ki = 44.2 nM T22939 C05VWL 122186744 Ki = 20.5 nM T22939 CNX5H4 122186745 Ki = 233 nM T22939 CQ6BG8 122186747 Ki = 5.51 nM T22939 CH8O2M 122186748 Ki = 86 nM T22939 C4LRN1 122186749 Ki = 29 nM T22939 CN9C2T 122192181 IC50 = 2691.53 nM T22939 C80TIN 122192182 IC50 > 31622.78 nM T22939 CZG5N9 122192183 IC50 = 724.44 nM T22939 CBE26N 122192184 IC50 = 1513.56 nM T22939 CP5ER0 122192185 IC50 = 33.11 nM T22939 CAR2M7 122192186 IC50 = 12.88 nM T22939 CZMK47 122192187 IC50 = 2290.87 nM T22939 CCP56N 122192188 IC50 = 48.98 nM T22939 C3KH0N 122192189 IC50 = 50.12 nM T22939 CI8KN0 122192190 IC50 = 3.631 nM T22939 C95FVG 122192191 IC50 = 0.8318 nM T22939 CCK36V 127029882 IC50 > 5000 nM T22939 CFY1P0 127029884 IC50 > 2000 nM T22939 CLDC46 127031152 IC50 > 37000 nM T22939 C60SMC 127031153 IC50 > 12000 nM T22939 CZET89 127050026 IC50 = 107 nM T22939 CPRJ71 127050027 IC50 = 26 nM T22939 CY0WZ9 129295280 IC50 = 3.4 nM T22939 C65RIZ 129295282 IC50 = 2488 nM T22939 CR23ZG 129295311 IC50 = 910 nM T22939 C2LVO7 129295370 IC50 = 4068 nM T22939 CTI04S 129295372 IC50 = 1640 nM T22939 C7MRB5 129304758 IC50 = 14.4 nM T22939 C12UNI 132502971 IC50 = 8000 nM T22939 C4GK7D 132578539 IC50 = 34 nM T22939 C0BZ5F 132578540 IC50 = 24 nM T22939 C4UFL6 134131799 IC50 = 270 nM T22939 C9YM8U 134133105 IC50 = 6000 nM T22939 C76DUH 134134996 IC50 = 250 nM T22939 CU5ZE0 134135805 IC50 = 650 nM T22939 C7Z6VF 134136082 IC50 = 850 nM T22939 CJ3D6N 134137415 IC50 = 290 nM T22939 C35USY 134137484 IC50 = 190 nM T22939 C9TG2N 134137487 IC50 = 794.33 nM T22939 COQG78 134138057 IC50 = 370 nM T22939 C28IKW 134138668 IC50 = 2200 nM T22939 C8KQ4M 134138731 IC50 = 38 nM T22939 C1SIE2 134139128 IC50 = 120 nM T22939 C36IYJ 134139595 IC50 = 550 nM T22939 C42MZI 134141921 IC50 = 480 nM T22939 CDW3L5 134141982 IC50 = 250 nM T22939 CF69JY 134142192 IC50 = 3800 nM T22939 C0WLC9 134143170 IC50 = 47 nM T22939 CRHX28 134143730 IC50 = 320 nM T22939 CN5M2S 134144292 IC50 = 2200 nM T22939 COGE75 134144424 IC50 = 450 nM T22939 CVS10N 134145032 IC50 = 210 nM T22939 CW8C6B 134145227 IC50 = 31 nM T22939 CK10EC 134145786 IC50 = 3000 nM T22939 CZ7DQ8 134146714 IC50 = 330 nM T22939 C9P3LQ 134146863 IC50 = 340 nM T22939 CH10EF 134148038 IC50 = 230 nM T22939 C7I2ZD 134148099 IC50 = 290 nM T22939 CSJV40 134148162 IC50 = 2600 nM T22939 C5VUQ6 134148654 IC50 = 570 nM T22939 CT59CV 134148906 IC50 = 15800 nM T22939 C0QJX4 134149670 IC50 = 230 nM T22939 C3PQM2 134149778 IC50 = 260 nM T22939 CI74TK 134149827 IC50 = 56 nM T22939 CML13S 134149996 IC50 = 150 nM T22939 C51AQU 134150642 IC50 = 140 nM T22939 CG8SY0 134150801 IC50 = 640 nM T22939 CU9C3R 134150891 IC50 = 190 nM T22939 C9C8GB 134151742 IC50 = 300 nM T22939 CA13RQ 134152665 IC50 = 450 nM T22939 CEFZ45 134153112 IC50 = 470 nM T22939 C3YD6S 134153484 IC50 = 440 nM T22939 C6MZK2 134154230 IC50 = 580 nM T22939 CR0TC6 134154275 IC50 = 2000 nM T22939 CC6DE5 134154860 IC50 = 220 nM T22939 CJ5Z7C 134154988 IC50 = 180 nM T22939 C87YMA 134156029 IC50 = 3500 nM T22939 CK2M5B 134156383 IC50 = 490 nM T22939 CW52PN 134157311 IC50 = 390 nM T22939 C1J6LN 134157750 IC50 = 160 nM T22939 C30HIQ 134415607 IC50 = 4.6 nM T22939 C3Y2NT 134415609 IC50 = 523 nM T22939 CQ53DW 134415610 IC50 = 4242 nM T22939 CO32XF 134415624 IC50 = 4.8 nM T22939 CRP1C4 134415742 IC50 = 21.1 nM T22939 C1U9HD 134415745 IC50 = 6 nM T22939 CB09XQ 134415864 IC50 = 527 nM T22939 CU6Y5D 134415868 IC50 = 25.4 nM T22939 CY8U6E 135459005 IC50 = 22500 nM T22939 CTF0J3 135567449 Ki = 2511.89 nM T22939 C34JMK 135571931 IC50 = 27700 nM T22939 C5MXO2 136000568 Ki = 27 nM T22939 CM6OX5 136000656 Ki = 950 nM T22939 C4K1XN 136045781 IC50 = 676.7 nM T22939 CZ2D6U 136059148 Ki = 220 nM T22939 C6HOU3 136059149 Ki = 570 nM T22939 CE1G9O 136059150 Ki = 3800 nM T22939 C7LSN6 136088946 Ki = 380 nM T22939 COI80Z 137634236 IC50 = 794.33 nM T22939 CPD87Y 137639726 IC50 = 630.96 nM T22939 C30ZJF 137648477 IC50 = 794.33 nM T22939 CO92KL 137654415 IC50 = 794.33 nM T22939 C7EKA2 138911324 IC50 = 1135 nM T22939 C96ONI 141538600 IC50 = 1689 nM T22939 CR6Y2I 141538601 IC50 = 1487 nM T22939 CW3Y0H 145949340 IC50 = 150 nM T22939 CEB89X 145949365 IC50 = 130 nM T22939 C9QUK1 145949374 IC50 = 1000 nM T22939 C4F0YC 145949647 IC50 = 210 nM T22939 CPK5U1 145951022 IC50 = 27 nM T22939 CKT24R 145951943 IC50 = 340 nM T22939 CGY64R 145955230 IC50 = 180 nM T22939 CIFB85 145957768 IC50 = 270 nM T22939 CS3N1H 145959892 IC50 = 310 nM T22939 CC7B4Q 145960034 IC50 = 360 nM T22939 C0Y4WE 145960285 IC50 = 730 nM T22939 C30SYM 155459658 IC50 = 2084 nM T22939 CGB78J 155459666 IC50 = 1546 nM T22939 C28RHM 155514304 Ki > 50118.72 nM T22939 CELU49 155517819 Ki > 50118.72 nM T22939 C2E4XV 155518137 Ki > 50118.72 nM T22939 C4QAB0 155518139 Ki > 50118.72 nM T22939 COF3R4 155520306 IC50 = 780 nM T22939 C1WAQ6 155527406 Ki = 25118.86 nM T22939 CB0XS4 155529625 Ki > 50118.72 nM T22939 C5Y4FK 155531943 IC50 > 1000 nM T22939 COP7X8 155539171 IC50 > 10000 nM T22939 C28KPU 155540268 IC50 > 1000 nM T22939 C1XGF5 155546726 IC50 = 8.2 nM T22939 CR5ZI2 155557239 Ki = 25118.86 nM T22939 C79WFJ 155567245 Ki > 50118.72 nM T22939 D00ZGW 46883841 IC50 = 1258.93 nM T22939 D01ETZ 261000 Ki = 0.49 nM T22939 D01NVD 46830196 IC50 = 3162.28 nM T22939 D02UID 16734800 IC50 > 1000 nM T22939 D02ZEE 25093227 IC50 = 3250 nM T22939 D04SAO 9799518 IC50 = 12.02 nM T22939 D05CND 10221123 IC50 = 83.8 nM T22939 D06DSF 24824217 IC50 = 300 nM T22939 D07KWO 9823099 IC50 = 2400 nM T22939 D07TVI 25093231 IC50 > 10000 nM T22939 D07XCB 17132382 IC50 = 11000 nM T22939 D08KQM 24816375 Ki = 866 nM T22939 D09OKK 9951771 Ki = 0.66 nM T22939 D09VWK 45483822 IC50 = 225 nM T22939 D0D6HI 46889764 IC50 = 224 nM T22939 D0E9CG 17067759 IC50 = 23000 nM T22939 D0F1SS 44605900 EC50 = 1.1 nM T22939 D0G5OV 11543746 IC50 = 4.1 nM T22939 D0GR5L 9906282 Ki = 1300 nM T22939 D0J7XZ 9819614 Ki > 10000 nM T22939 D0L5IC 9820558 Ki > 10000 nM T22939 D0M0RS 11560224 Ki > 1000 nM T22939 D0N1RQ 15908132 IC50 = 103 nM T22939 D0V4PL 9903358 IC50 = 27 nM T22939 D0V4RZ 25113722 IC50 > 10000 nM T22939 D0V9NE 4369524 EC50 = 0.15 nM T22939 D0XS0R 44433505 Ki = 29424 nM T22939 D0ZM6R 77098 Ki = 131.83 nM T76508 D0E3TC 44259 IC50 = 43.5 nM T76508 C3VRO9 44557921 IC50 > 10000 nM T76508 CV63UL 67240318 IC50 > 10000 nM T76508 CXC69T 137321158 IC50 = 255 nM T76508 CS61AX 137659496 IC50 > 100000 nM T76508 CM3A8O 139030333 IC50 = 910 nM T76508 C6VB3O 145925651 IC50 = 2200 nM T76508 C2MD1Q 155513187 IC50 > 10000 nM T76508 CC9LQ2 155546287 IC50 = 5800 nM T76508 D07ADX 54764565 IC50 = 661 nM T78356 D0C7AA 5282440 IC50 = 24 nM T78356 D0E3BH 5362391 IC50 = 3 nM T78356 D0M6DO 2145 IC50 = 18500 nM T78356 D0R1RS 3715 IC50 = 100 nM T78356 D0D9LB 6449876 IC50 = 4 nM T78356 D04EEU 53001 IC50 = 3 nM T78356 D07JSK 51550 IC50 = 94100 nM T78356 D09DIG 57109 IC50 = 6000 nM T78356 D09QRO 55390 IC50 = 3 nM T78356 D0H5PG 131717 IC50 = 2 nM T78356 D0JY4Y 443292 IC50 = 9 nM T78356 D0K4UW 65922 IC50 = 6 nM T78356 D0OO6A 5284442 IC50 = 0.89 nM T78356 CF06EN 795 IC50 = 670000 nM T78356 CWV0R6 53000 IC50 = 14 nM T78356 C7I6HX 53555 IC50 = 28 nM T78356 C9T3FB 105007 IC50 = 10000 nM T78356 C1WGZ7 119553 IC50 = 12 nM T78356 CW45IU 126253 IC50 = 150 nM T78356 C1JP9N 129519 IC50 = 2 nM T78356 CAH01V 131713 IC50 = 210 nM T78356 CAS0I7 134834 IC50 = 9900 nM T78356 C7ZI5R 173117 IC50 = 39 nM T78356 C2G7SL 192280 IC50 = 1600 nM T78356 CK7TE9 192281 IC50 = 500 nM T78356 CGR38C 193906 IC50 = 400 nM T78356 CVJ1L9 368695 IC50 = 1100 nM T78356 CUE37L 3077003 IC50 = 2 nM T78356 COC2U7 3078928 IC50 = 24000 nM T78356 C5B4DK 4519262 IC50 = 2000 nM T78356 C5IA3R 6365736 IC50 = 3 nM T78356 CY4N6E 6436053 IC50 = 4 nM T78356 CA6V8C 6438130 IC50 = 11 nM T78356 CO2F7E 6439492 IC50 = 19 nM T78356 C0NQ7I 6450501 IC50 > 100000 nM T78356 CM2B0C 6537201 IC50 = 0.9 nM T78356 CV75GZ 6537211 IC50 = 490 nM T78356 C89XMB 6604763 IC50 > 100000 nM T78356 CU1MC9 9803080 IC50 = 1 nM T78356 CT02HX 9816806 IC50 = 30 nM T78356 CX8RM2 9830229 IC50 = 31.62 nM T78356 C6XP8J 9869582 IC50 = 18 nM T78356 CJ9E7N 9921473 IC50 = 32 nM T78356 CGT56V 9930263 IC50 = 380 nM T78356 C3L8VN 9940231 IC50 = 65 nM T78356 CS0HT9 9958626 IC50 = 55 nM T78356 CVF6Q2 9972369 IC50 = 120 nM T78356 CJ37ZT 9978095 IC50 = 77 nM T78356 CAHW97 9978952 IC50 > 500 nM T78356 CZQ0O9 9979675 IC50 = 24 nM T78356 C4TV0E 9982645 IC50 = 4 nM T78356 CDM12O 9983481 IC50 = 45000 nM T78356 CR2JK5 9997733 IC50 = 54 nM T78356 CH2WT0 10000478 IC50 = 50 nM T78356 CVU8B4 10002506 IC50 = 240 nM T78356 C7P9MS 10002804 IC50 = 5 nM T78356 C76HXM 10005561 IC50 = 39 nM T78356 C01XRG 10005641 IC50 = 2 nM T78356 CD9KR1 10008231 IC50 > 10000 nM T78356 CSK8U0 10010367 IC50 = 70 nM T78356 C3H4XZ 10010816 IC50 > 10000 nM T78356 C2HF1M 10025569 IC50 = 40 nM T78356 C3TVW4 10027568 IC50 = 1 nM T78356 CUO4P3 10028328 IC50 = 4 nM T78356 C81NMY 10031827 IC50 = 50 nM T78356 C7USV6 10032304 IC50 = 30 nM T78356 C5Y0MK 10036693 IC50 = 630 nM T78356 C5FH9Q 10047212 IC50 = 220 nM T78356 CH3W6U 10047870 IC50 = 2700 nM T78356 CK6S8D 10048962 IC50 = 3 nM T78356 CS63TX 10049649 IC50 = 18 nM T78356 CF1U8M 10050297 IC50 = 4 nM T78356 CY8JL4 10050856 IC50 = 20 nM T78356 CW8MU3 10051348 IC50 = 19 nM T78356 C9YBV0 10052055 IC50 = 5 nM T78356 C09LFU 10052612 IC50 = 25 nM T78356 CPCT06 10055313 IC50 = 20 nM T78356 CWB7K1 10055372 IC50 = 10 nM T78356 CZW7P4 10067523 IC50 = 6 nM T78356 C86HNP 10068983 IC50 = 200 nM T78356 CM86KR 10072535 IC50 = 60 nM T78356 C84PMW 10072583 IC50 = 5 nM T78356 CRC31H 10072780 IC50 = 5 nM T78356 CSXK61 10073256 IC50 = 100 nM T78356 C9U8FV 10073846 IC50 = 850 nM T78356 C6B0RS 10074652 IC50 = 24 nM T78356 C2MIC0 10074653 IC50 = 33 nM T78356 C9KP4Y 10075114 IC50 = 44 nM T78356 CP68RF 10075294 IC50 = 6 nM T78356 CYR5U6 10077517 IC50 = 30 nM T78356 C2L3XW 10078249 IC50 = 10 nM T78356 CLPO31 10078486 IC50 = 30 nM T78356 CP19IX 10091054 IC50 = 20 nM T78356 C1RVW5 10091337 IC50 = 2000 nM T78356 CYJX29 10093645 IC50 = 120 nM T78356 CS1Y8A 10094462 IC50 = 830 nM T78356 CK9F3Y 10095579 IC50 = 1400 nM T78356 CGBH15 10095993 IC50 = 5 nM T78356 CV4TL1 10096378 IC50 = 98 nM T78356 C7H1AI 10096697 IC50 = 5 nM T78356 CDG29R 10100855 IC50 = 60 nM T78356 CQI61A 10101127 IC50 = 30 nM T78356 CN3ZG5 10101171 IC50 = 50 nM T78356 C8NEV0 10101297 IC50 = 50 nM T78356 CEN72F 10243493 IC50 = 1600 nM T78356 C45WPL 10246884 IC50 = 100 nM T78356 C1M7SL 10252930 IC50 = 40 nM T78356 CTH17D 10253167 IC50 = 70 nM T78356 CR8FQ7 10253361 IC50 = 4.5 nM T78356 C3CU7G 10254161 IC50 = 7 nM T78356 CLMR13 10254162 IC50 = 21 nM T78356 CN6Z5J 10254246 IC50 = 38 nM T78356 CNZI93 10254733 IC50 = 39 nM T78356 C3SO9M 10255332 IC50 = 250 nM T78356 CGS2U4 10256828 IC50 = 310 nM T78356 CQO10R 10257045 IC50 = 1700 nM T78356 CJ2UC5 10257263 IC50 = 20 nM T78356 CD04FL 10258317 IC50 = 46 nM T78356 C6YW4C 10258999 IC50 = 40 nM T78356 CY32FE 10259965 IC50 > 10000 nM T78356 CUE72P 10314633 IC50 = 2500 nM T78356 CT7K8Z 10320386 IC50 = 21 nM T78356 C81XIN 10321242 IC50 = 20000 nM T78356 CCX54V 10321666 IC50 = 48 nM T78356 CVB78G 10321764 IC50 = 2.6 nM T78356 CDI40A 10321942 IC50 = 39 nM T78356 CEZA10 10321974 IC50 = 4 nM T78356 C4MLU9 10322324 IC50 = 3 nM T78356 CVQ6W7 10323516 IC50 = 61 nM T78356 C1KHU2 10327444 IC50 = 40 nM T78356 CGS16O 10327581 IC50 = 40 nM T78356 CN93TI 10327694 IC50 = 20 nM T78356 C50TPZ 10327812 IC50 = 21 nM T78356 CC1UF0 10335738 IC50 = 810 nM T78356 CKAU36 10343670 IC50 = 43 nM T78356 CI9Z5V 10343973 IC50 = 13 nM T78356 CQE7L9 10345903 IC50 = 31 nM T78356 C95HPE 10347272 IC50 = 150 nM T78356 CH0L6C 10359399 IC50 = 450 nM T78356 CK1Q7G 10359400 IC50 = 17000 nM T78356 C8JB2A 10361347 IC50 = 4 nM T78356 CJU03S 10367365 IC50 = 1.5 nM T78356 C1UD9O 10367382 IC50 = 3 nM T78356 CWR7X9 10369102 IC50 = 8 nM T78356 CK87GB 10369704 IC50 = 19 nM T78356 CWZ14V 10370098 IC50 = 5 nM T78356 CK23JW 10371334 IC50 = 4 nM T78356 CV59MZ 10372661 IC50 = 40 nM T78356 C78LHO 10382877 IC50 = 1900 nM T78356 CX53ZT 10384315 IC50 = 6100 nM T78356 CJ1QE0 10385168 IC50 = 693 nM T78356 C6ZWI7 10388467 IC50 = 7 nM T78356 C1TF0X 10389298 IC50 = 370 nM T78356 C5CRJ2 10391135 IC50 = 4 nM T78356 CPE5C2 10394030 IC50 = 30 nM T78356 CHNR09 10407142 IC50 > 10000 nM T78356 CT1P0N 10410915 IC50 = 20 nM T78356 C2BEN5 10411480 IC50 = 5 nM T78356 CFWJ57 10412393 IC50 = 2200 nM T78356 COW49N 10417774 IC50 = 41 nM T78356 C25MYB 10425738 IC50 = 390 nM T78356 CCN15P 10429343 IC50 = 9 nM T78356 CGZ80R 10431466 IC50 = 940 nM T78356 C9XH6A 10432271 IC50 > 10000 nM T78356 C5OGH6 10432964 IC50 = 1 nM T78356 CQG62B 10434230 IC50 = 7 nM T78356 C4GDE3 10436457 IC50 = 4 nM T78356 CZ82UL 10438021 IC50 = 40 nM T78356 CDB71L 10438679 IC50 = 60 nM T78356 C8WKX9 10451585 IC50 = 16 nM T78356 C9B3TD 10455364 IC50 = 40000 nM T78356 CA1L8E 10456329 IC50 = 3 nM T78356 CFY19A 10457312 IC50 = 150 nM T78356 C85KTH 10457484 IC50 = 4 nM T78356 C0X3OS 10458951 IC50 = 21 nM T78356 CKIH16 10460371 IC50 = 100 nM T78356 CH9Y2F 10460682 IC50 > 10000 nM T78356 CA4S6T 10462005 IC50 = 30 nM T78356 C7IL0E 10462692 IC50 = 72 nM T78356 CT1U9V 10475510 IC50 > 10000 nM T78356 CSP02I 10478324 IC50 = 70 nM T78356 CY27WV 10478768 IC50 = 14 nM T78356 CJCL19 10479578 IC50 = 5 nM T78356 C7RJ5Y 10479865 IC50 = 5 nM T78356 CJ2T5E 10483231 IC50 = 43 nM T78356 CG3IB6 10484455 IC50 = 10 nM T78356 CY73UJ 10485192 IC50 = 20 nM T78356 C9W6YH 10488782 IC50 = 2000 nM T78356 CYR2O4 10489655 IC50 = 1700 nM T78356 CU90BJ 10494367 IC50 > 100000 nM T78356 C9L1JY 10500482 IC50 = 22 nM T78356 CA8CF2 10500543 IC50 = 3900 nM T78356 CL76FX 10502084 IC50 = 22 nM T78356 C60WMU 10503252 IC50 = 320 nM T78356 C68XED 10503638 IC50 = 930 nM T78356 C27HCL 10504682 IC50 = 38 nM T78356 C20LIQ 10505899 IC50 = 2.6 nM T78356 CH2R0N 10513661 IC50 = 1260 nM T78356 C18NWE 10518243 IC50 > 100000 nM T78356 C3TY0D 10518244 IC50 > 100000 nM T78356 CUFL39 10524500 IC50 = 24 nM T78356 C9IU3F 10526115 IC50 = 6 nM T78356 C3XID0 10526677 IC50 = 3 nM T78356 C3ZB8E 10530889 IC50 = 11.5 nM T78356 CBPQ89 10542153 IC50 = 8800 nM T78356 C54MEV 10543197 IC50 = 3800 nM T78356 CUC93I 10545734 IC50 = 430 nM T78356 CF4G6L 10548488 IC50 = 400 nM T78356 CM3AW2 10549479 IC50 = 48 nM T78356 CW73IA 10550018 IC50 = 3 nM T78356 C5NWI6 10551940 IC50 = 37 nM T78356 C2C1VJ 10552843 IC50 = 3 nM T78356 C7RH0M 10554248 IC50 = 36.7 nM T78356 C2A6CY 10554249 IC50 = 42 nM T78356 CP4XJ9 10576417 IC50 = 54 nM T78356 C7S5RV 10586086 IC50 = 680 nM T78356 CRU0P1 10591274 IC50 > 10000 nM T78356 CD1V5X 10601327 IC50 = 4 nM T78356 CA6J2P 10601707 IC50 = 5.9 nM T78356 CDXM71 10602360 IC50 = 63 nM T78356 C3DH9W 10608774 IC50 = 1010 nM T78356 CQ0PC7 10619606 IC50 = 26 nM T78356 CZT9C2 10620837 IC50 = 22 nM T78356 C8SRW4 10626384 IC50 = 28.7 nM T78356 CEC6Q0 10637870 IC50 = 260 nM T78356 CH1VS3 10637871 IC50 = 75 nM T78356 CD53UC 10648075 IC50 = 53 nM T78356 C19HPG 10649580 IC50 = 50.8 nM T78356 CX1R3B 10661867 IC50 = 620 nM T78356 CGRY48 10669025 IC50 = 4 nM T78356 C4NGP3 10669026 IC50 = 25 nM T78356 CUD90Y 10669649 IC50 = 3 nM T78356 CM54YJ 10669723 IC50 = 39 nM T78356 CN05QE 10670440 IC50 = 5 nM T78356 CKXG92 10670672 IC50 = 37 nM T78356 CP98RW 10680142 IC50 = 4100 nM T78356 CYGK01 10686657 IC50 > 10000 nM T78356 CL8OZ7 10686658 IC50 > 10000 nM T78356 C8JW6U 10696378 IC50 = 61 nM T78356 C0K1ZP 10697301 IC50 = 3 nM T78356 CT14ZS 10717572 IC50 = 180 nM T78356 C6DPF4 10717914 IC50 = 11 nM T78356 C4Y2AP 10720045 IC50 = 9.4 nM T78356 C4TE6Y 10728303 IC50 = 2000 nM T78356 C1ICD7 10741449 IC50 = 230 nM T78356 C28ETW 10742084 IC50 = 38 nM T78356 C50QCV 10744075 IC50 = 49 nM T78356 CU5W7P 10752634 IC50 = 2300 nM T78356 C3QZJ8 10756559 IC50 = 573 nM T78356 C1PHY8 10756560 IC50 > 100000 nM T78356 C53NGA 10756561 IC50 = 79 nM T78356 CM51CL 10761205 IC50 = 250 nM T78356 CMF5P7 10762387 IC50 > 10000 nM T78356 CTBF04 10762411 IC50 = 4 nM T78356 CVQ3J9 10764618 IC50 = 2900 nM T78356 C3AJ5O 10764758 IC50 = 200 nM T78356 C0FCK3 10764803 IC50 = 45 nM T78356 C7N0GM 10765092 IC50 = 43 nM T78356 C17OLN 10766313 IC50 = 25 nM T78356 C5QN7D 10768214 IC50 = 33 nM T78356 C03YOG 10768772 IC50 = 48.9 nM T78356 CZIW89 10768926 IC50 = 49 nM T78356 C2GML0 10769084 IC50 = 49.2 nM T78356 CCD9R4 10774996 IC50 = 3550 nM T78356 C4AB0L 10780482 IC50 > 10000 nM T78356 CF5E4M 10786712 IC50 = 3900 nM T78356 CL9QH2 10789321 IC50 = 20 nM T78356 CE9D3P 10810477 IC50 = 22 nM T78356 C0EAP2 10823139 IC50 = 3400 nM T78356 C8CV6J 10827996 IC50 > 100000 nM T78356 CXZ15O 10833696 IC50 > 10000 nM T78356 CUL9A6 10834261 IC50 = 29 nM T78356 CE3J4M 10835548 IC50 = 18 nM T78356 CEZ8D1 10840154 IC50 = 2.7 nM T78356 CU3I7B 10847200 IC50 = 1230 nM T78356 CTOQ40 10852668 IC50 > 10000 nM T78356 COK72V 11171316 IC50 > 1000 nM T78356 C1OV2B 11480797 IC50 = 500 nM T78356 C2XQI7 11526708 IC50 = 950 nM T78356 C45NBF 11705274 IC50 = 800 nM T78356 CZ7J3P 11743126 IC50 > 10000 nM T78356 CP78LQ 11744722 IC50 = 3.5 nM T78356 C5LMZ4 11753841 IC50 = 1000 nM T78356 CZ5J9I 11754506 IC50 = 2 nM T78356 C9LXS2 11754856 IC50 = 15000 nM T78356 CM3B0K 11755215 IC50 = 60 nM T78356 CXW63P 11755659 IC50 = 15 nM T78356 CT14SM 11796350 IC50 = 29 nM T78356 CP05GO 11796543 IC50 = 27 nM T78356 C9L1SP 11796683 IC50 = 38 nM T78356 CSG2U1 11796949 IC50 = 43 nM T78356 CJ42SC 11800240 IC50 = 47.5 nM T78356 C20VHX 12803314 IC50 > 1000 nM T78356 CFP3K8 12870347 IC50 = 20000 nM T78356 CVF4E0 12870354 IC50 = 20000 nM T78356 C0TIZ7 12870387 IC50 = 134 nM T78356 CN58PQ 12870425 IC50 = 32 nM T78356 CPZ47L 12870426 IC50 = 30 nM T78356 CV8YW3 12870428 IC50 = 46 nM T78356 CZLH92 12870430 IC50 = 140 nM T78356 C09FWG 12870432 IC50 = 250 nM T78356 C90JKU 12870434 IC50 = 1500 nM T78356 C39SDO 12870436 IC50 = 44 nM T78356 C32LJO 12870438 IC50 = 1600 nM T78356 CLG51X 12870440 IC50 = 4 nM T78356 C2ISR9 12870442 IC50 = 250 nM T78356 C9CME6 12870444 IC50 = 31 nM T78356 C2FZ4P 12870445 IC50 = 40 nM T78356 CPLX68 12870446 IC50 = 210 nM T78356 CQO26U 12870448 IC50 = 38 nM T78356 C9F4PQ 12870450 IC50 = 25 nM T78356 CBQ5L2 12870452 IC50 = 95 nM T78356 CNER79 12870454 IC50 = 30 nM T78356 CN7ER2 12870456 IC50 = 42 nM T78356 CCX19R 12870458 IC50 = 120 nM T78356 CC6UO2 12870460 IC50 = 42 nM T78356 CVC4I0 12870462 IC50 = 70 nM T78356 C31VAR 12870464 IC50 = 16 nM T78356 C2QY8C 12870466 IC50 = 30 nM T78356 C9E4VG 12870468 IC50 = 9 nM T78356 C3EWY4 12870470 IC50 > 1000 nM T78356 C0MIJ3 12870471 IC50 = 16 nM T78356 C9LNJ8 12870482 IC50 = 450 nM T78356 CCX4R3 12870484 IC50 = 40 nM T78356 C5S1EQ 12870486 IC50 = 53 nM T78356 C31NIC 12870495 IC50 = 90 nM T78356 C0A7KB 12870497 IC50 = 71 nM T78356 CO4KB6 12870499 IC50 = 54 nM T78356 CUME96 12870503 IC50 = 56 nM T78356 CD9HE3 12870509 IC50 = 25 nM T78356 COLS61 12870511 IC50 > 1000 nM T78356 CO2BR5 12870524 IC50 = 5 nM T78356 CJ2O4Y 12870528 IC50 >> 1000 nM T78356 C52ATC 12870529 IC50 = 1200 nM T78356 C6L9MV 12870534 IC50 = 3300 nM T78356 CPH87C 12870537 IC50 = 38 nM T78356 COG56Z 12870540 IC50 = 550 nM T78356 CK39LO 12882185 IC50 = 210 nM T78356 C2H7SI 12882187 IC50 = 10 nM T78356 C29BLK 12882190 IC50 = 20 nM T78356 CO5C7H 12882192 IC50 = 5 nM T78356 CS7CN6 12882198 IC50 = 7 nM T78356 C40DZF 12904547 IC50 = 68 nM T78356 CPN68W 12904549 IC50 > 1000 nM T78356 C2TLN5 12904560 IC50 = 86 nM T78356 CCX20D 12904562 IC50 > 1000 nM T78356 CUN0J2 12904564 IC50 = 76 nM T78356 CC3IV6 12904566 IC50 > 1000 nM T78356 CWH60T 12904577 IC50 = 56 nM T78356 C60MTP 12904585 IC50 = 47 nM T78356 C3FMO9 12904587 IC50 = 12 nM T78356 CU0GM8 12904593 IC50 = 25 nM T78356 C46NOW 12904603 IC50 > 1000 nM T78356 CFJ3L6 13094289 IC50 = 70 nM T78356 C6DHP4 13206138 IC50 = 330 nM T78356 C4X0NS 13206139 IC50 = 5.2 nM T78356 CQ21UW 13206140 IC50 = 21 nM T78356 CCI3G1 13206142 IC50 = 41 nM T78356 CO6XW4 13206143 IC50 = 77 nM T78356 CM14UX 13206144 IC50 = 270 nM T78356 CDH35G 13206145 IC50 = 550 nM T78356 CI6Q2S 13206146 IC50 = 280 nM T78356 CRI0Z3 13206149 IC50 = 4.8 nM T78356 C9LIT8 13206150 IC50 = 40 nM T78356 CGWC95 13206151 IC50 = 390 nM T78356 C46DXA 13206152 IC50 = 3300 nM T78356 CJ89OX 13206153 IC50 = 4700 nM T78356 CD3EZ1 13206156 IC50 = 28 nM T78356 CF16NP 13206159 IC50 = 25000 nM T78356 CX2WQ8 13285828 IC50 = 85 nM T78356 C9TFL1 13285829 IC50 = 19 nM T78356 C1PHM2 13285830 IC50 = 60 nM T78356 C42KLH 13285831 IC50 = 41 nM T78356 CW83DY 13285832 IC50 = 56 nM T78356 CCA0S5 13285833 IC50 = 20 nM T78356 CCHY95 13285834 IC50 = 54 nM T78356 CP5IO2 13285851 IC50 = 1300 nM T78356 C86WIL 13322231 IC50 = 34 nM T78356 CP0G5X 13373631 IC50 = 11 nM T78356 CMN13Q 13373633 IC50 = 19 nM T78356 CEC3R6 13373634 IC50 = 20 nM T78356 CHT62M 13417256 IC50 = 450 nM T78356 C9RWK8 13417257 IC50 = 110 nM T78356 CCI6Y5 13417258 IC50 = 280 nM T78356 CMC39D 13417259 IC50 = 65 nM T78356 CZNC95 13417260 IC50 = 29 nM T78356 C05QNE 13417262 IC50 = 230 nM T78356 CPVG63 13417263 IC50 = 32 nM T78356 C0OYX5 13417264 IC50 = 310 nM T78356 CRZM34 13417265 IC50 = 42 nM T78356 CG6Q4M 13417266 IC50 = 520 nM T78356 CAM6Q2 13417267 IC50 = 55 nM T78356 C4XNE9 13417268 IC50 = 2700 nM T78356 C2I1MU 13417269 IC50 > 100000 nM T78356 CZ0V3J 13417273 IC50 = 130 nM T78356 CFR6U1 13417276 IC50 = 70 nM T78356 C75QFY 13417277 IC50 = 52 nM T78356 C81WQV 13417278 IC50 = 73 nM T78356 C9DG0P 13417280 IC50 = 210 nM T78356 CQU68F 13417281 IC50 = 71 nM T78356 CHCF69 13417284 IC50 = 34 nM T78356 C3AH9B 13417285 IC50 = 31 nM T78356 CD1XY7 13417286 IC50 = 62 nM T78356 C5TUO0 13417289 IC50 = 980 nM T78356 CB45QK 13417290 IC50 = 100 nM T78356 CF1KS6 13417291 IC50 = 30 nM T78356 CH9O1L 13417292 IC50 = 21 nM T78356 C7JW6Y 13417293 IC50 = 38 nM T78356 C8UEW4 13417294 IC50 = 45 nM T78356 COX4L0 13417295 IC50 = 37 nM T78356 CQZR39 13417296 IC50 = 18 nM T78356 C6GK5T 13417297 IC50 = 43 nM T78356 CAN15O 13417298 IC50 = 48 nM T78356 CAWN72 13417299 IC50 = 50 nM T78356 CIUH27 13417300 IC50 = 32 nM T78356 CT4R8D 13417302 IC50 = 100 nM T78356 CBG52Y 13417304 IC50 = 600 nM T78356 CW7KX5 13417306 IC50 = 33 nM T78356 C3DT6W 13417308 IC50 = 30 nM T78356 C2G1IF 13417310 IC50 = 110 nM T78356 C8M5IB 13417312 IC50 = 58 nM T78356 C23TFI 13417314 IC50 = 50 nM T78356 C6NKO1 13417316 IC50 = 28 nM T78356 CY96AW 13417317 IC50 = 65 nM T78356 C7I5GY 13417319 IC50 = 42 nM T78356 CB52NE 13417321 IC50 = 41 nM T78356 CFM8E0 13417323 IC50 = 60 nM T78356 C7BE9J 13417325 IC50 = 28 nM T78356 C1T8EJ 13417327 IC50 = 2200 nM T78356 C5WQU0 13417329 IC50 = 400 nM T78356 C1BX3E 13417330 IC50 > 10000 nM T78356 CGD2P5 13557455 IC50 = 100 nM T78356 C4TLY1 13557457 IC50 = 4000 nM T78356 C9DH8J 13557459 IC50 = 100 nM T78356 CH93FQ 13557460 IC50 = 200 nM T78356 C16UNF 13557463 IC50 = 100 nM T78356 C8LYE5 13557464 IC50 = 50 nM T78356 CGKW06 13557472 IC50 = 100 nM T78356 C2AG1U 13557473 IC50 = 200 nM T78356 C1X0ZV 13557474 IC50 = 60 nM T78356 C8FUQ7 13557475 IC50 = 20 nM T78356 C6PO3S 13557476 IC50 = 100 nM T78356 CBF1U7 13557477 IC50 = 60 nM T78356 C4VSK3 13557479 IC50 > 10000 nM T78356 CO6MT9 13557480 IC50 = 600 nM T78356 C6XHY0 13557482 IC50 = 200 nM T78356 CS65WV 13557485 IC50 = 5000 nM T78356 C70OND 13557486 IC50 = 200 nM T78356 CZP63Y 13557492 IC50 = 600 nM T78356 C6UCY3 13557494 IC50 = 20 nM T78356 CD6LE3 13557495 IC50 = 20 nM T78356 CQ7AP9 13557497 IC50 = 100 nM T78356 CHG45B 13557498 IC50 = 300 nM T78356 C03AUE 13557505 IC50 = 1000 nM T78356 CQ8L5Y 13569173 IC50 = 4400 nM T78356 CM23VB 13569174 IC50 = 22000 nM T78356 CT1ZL2 13569175 IC50 = 2000 nM T78356 CLOP75 13569178 IC50 = 2900 nM T78356 CSY2V4 13569179 IC50 = 1800 nM T78356 CU69WY 13569180 IC50 = 610 nM T78356 C86EAW 13569181 IC50 = 3000 nM T78356 CM3UA6 13569183 IC50 = 3500 nM T78356 C4BT5G 13569185 IC50 = 4000 nM T78356 CB3X2Y 13569186 IC50 > 50000 nM T78356 CH1I6N 13569187 IC50 > 10000 nM T78356 C1VNT2 13569189 IC50 > 10000 nM T78356 CE01PH 13569191 IC50 = 95 nM T78356 CPWB08 13569193 IC50 = 32 nM T78356 CC07NV 13569194 IC50 = 530 nM T78356 C37HVK 13569196 IC50 = 860 nM T78356 C4GRJ1 13569197 IC50 = 1100 nM T78356 CH7K9W 13569198 IC50 = 13000 nM T78356 CCB9W8 13569199 IC50 = 15 nM T78356 CZ75ML 13569200 IC50 = 630 nM T78356 C4L3HD 13569201 IC50 = 180 nM T78356 CIA14L 13569202 IC50 = 850 nM T78356 CA6F4K 13569203 IC50 > 5000 nM T78356 CQ9A0D 13569204 IC50 = 840 nM T78356 CN48UY 13569205 IC50 > 50000 nM T78356 CL3W9U 13590268 IC50 = 560 nM T78356 C7F5PR 13594137 IC50 = 3000 nM T78356 CV37RZ 13594138 IC50 = 4600 nM T78356 CCAN10 13594154 IC50 = 30 nM T78356 CCF4E0 13594155 IC50 = 19 nM T78356 C4GR2M 13594156 IC50 = 8.2 nM T78356 C5EI9O 13594158 IC50 = 42 nM T78356 CB94PC 13594159 IC50 = 43 nM T78356 C39EWI 13594160 IC50 = 21 nM T78356 C3NV6O 13594161 IC50 = 12 nM T78356 C61EUC 13594162 IC50 = 82 nM T78356 C4CIL0 13594163 IC50 = 10 nM T78356 CY06BU 13663018 IC50 = 20 nM T78356 C2RO1K 13663020 IC50 = 18 nM T78356 CA2G0U 13663021 IC50 = 19 nM T78356 C4B0JT 13663022 IC50 = 5.2 nM T78356 C4ZL3M 13663023 IC50 = 7.4 nM T78356 CTO6Q2 13663024 IC50 = 5 nM T78356 C3LTJ0 13663025 IC50 = 52 nM T78356 CSA28P 13663026 IC50 = 21 nM T78356 C3I0PO 13663027 IC50 = 1700 nM T78356 CF65LR 13663028 IC50 = 29 nM T78356 CP3YJ0 13663029 IC50 = 120 nM T78356 CERG39 13663030 IC50 = 34 nM T78356 C8D7GL 13663031 IC50 = 5 nM T78356 C1GR7Q 13663032 IC50 = 33 nM T78356 C52TQH 13663033 IC50 = 420 nM T78356 CA73JR 13663034 IC50 = 140 nM T78356 CF8Y2B 13663089 IC50 = 12 nM T78356 CLA7H9 13663090 IC50 = 34 nM T78356 CBL5S7 13663091 IC50 = 31 nM T78356 C5Y3SG 13663092 IC50 = 30 nM T78356 C2Y5SB 13663093 IC50 = 15 nM T78356 C2A5FS 13663094 IC50 = 17 nM T78356 C6XU4Y 13663096 IC50 = 18 nM T78356 CPFG92 13663097 IC50 = 40 nM T78356 CYED42 13663098 IC50 = 22 nM T78356 CC35VH 13663099 IC50 = 27 nM T78356 CF3Y4H 13663100 IC50 = 43 nM T78356 CUQC45 13663101 IC50 = 37 nM T78356 C2EL3W 13663102 IC50 = 32 nM T78356 CR8WH0 13663104 IC50 = 34 nM T78356 C8E4PJ 13739736 IC50 = 500 nM T78356 C4TF2D 13739744 IC50 = 300 nM T78356 CDT5E9 13750120 IC50 = 27 nM T78356 C4JZ6M 13904791 IC50 = 730 nM T78356 CWT6I0 13904792 IC50 = 1890 nM T78356 C82DLP 13904793 IC50 = 120 nM T78356 C8ZDM0 13904794 IC50 = 420 nM T78356 CXV3F0 13904795 IC50 = 36 nM T78356 CRD69G 13904796 IC50 > 20000 nM T78356 CM4TX3 13904802 IC50 = 390 nM T78356 CM18DE 13904804 IC50 = 17600 nM T78356 C86BWG 13904805 IC50 = 1430 nM T78356 C03JNE 13904806 IC50 = 120 nM T78356 CIJ13P 13904807 IC50 = 750 nM T78356 CP8LY3 13904808 IC50 = 4000 nM T78356 C04XGV 13904809 IC50 = 1000 nM T78356 CH9N6B 13904812 IC50 = 10000 nM T78356 CI4L6S 13904813 IC50 = 8330 nM T78356 C7A3FU 13904989 IC50 = 1260 nM T78356 CZ72MO 13904990 IC50 = 540 nM T78356 CN8A9P 13904991 IC50 = 6400 nM T78356 CJ4K9U 13904994 IC50 = 3600 nM T78356 C3P9RW 13904995 IC50 = 700 nM T78356 C3RFB6 13904996 IC50 = 7200 nM T78356 CR0G9Y 13904997 IC50 = 6200 nM T78356 CX57WK 13904998 IC50 = 8600 nM T78356 CL3GD8 13904999 IC50 = 180 nM T78356 C5DX6I 13905000 IC50 = 1610 nM T78356 C39ZWY 13905001 IC50 = 200 nM T78356 C9HW6M 13905002 IC50 = 560 nM T78356 C9L3SC 13905003 IC50 = 1490 nM T78356 C56CJR 13905004 IC50 = 21000 nM T78356 CEU01T 13905005 IC50 = 6000 nM T78356 CIN16O 13905006 IC50 = 12400 nM T78356 C0QM6R 13905007 IC50 = 1940 nM T78356 CF6R8S 13905008 IC50 = 5400 nM T78356 C4DKS2 13905009 IC50 = 24900 nM T78356 C70PWB 13905010 IC50 = 12400 nM T78356 C48TMW 13937678 IC50 = 93 nM T78356 CBU93K 13937680 IC50 = 86 nM T78356 CTC6S0 13937687 IC50 = 100 nM T78356 CG63QO 13952788 IC50 = 10 nM T78356 COC0I3 14071622 IC50 = 26 nM T78356 CBI82L 14277789 IC50 = 490 nM T78356 C69RCW 14373260 IC50 = 350 nM T78356 CE7L8R 14373269 IC50 = 1200 nM T78356 CB41NR 14373278 IC50 = 25000 nM T78356 CKA2T4 14501917 IC50 = 114 nM T78356 C7EAX6 14501929 IC50 = 2680 nM T78356 C74ZGI 14501941 IC50 = 1850 nM T78356 CSB0K8 14501965 IC50 > 10000 nM T78356 CF0PE7 14501968 IC50 > 10000 nM T78356 CM3SF6 14501971 IC50 = 114 nM T78356 C4YCK1 14501992 IC50 > 10000 nM T78356 C8CT4D 14820371 IC50 = 1 nM T78356 CJ64MH 14820372 IC50 = 1 nM T78356 C4GRH3 14986630 IC50 > 1000 nM T78356 CEG92V 14986636 IC50 = 90 nM T78356 CE6B1W 14986638 IC50 = 10 nM T78356 C54OGM 15024085 IC50 = 630.96 nM T78356 C5N6JP 15024086 IC50 = 100 nM T78356 C1MAW4 15024087 IC50 = 2511.89 nM T78356 CH47DU 15024088 IC50 = 100 nM T78356 CE4Z0F 15024089 IC50 = 100 nM T78356 C5ZEO4 15024090 IC50 < 10000 nM T78356 CNY9T8 15024091 IC50 = 1584.89 nM T78356 CXTV01 15024092 IC50 < 10000 nM T78356 C6S1XA 15024093 IC50 < 10000 nM T78356 CYLC70 15024094 IC50 < 10000 nM T78356 C36SHE 15024095 IC50 = 630.96 nM T78356 C1MF5W 15024096 IC50 < 10000 nM T78356 C4F5UH 15024097 IC50 = 1584.89 nM T78356 CK6RS0 15024098 IC50 = 398.11 nM T78356 CA85FM 15290511 IC50 = 210000 nM T78356 C63ZRQ 15290512 IC50 > 1000000 nM T78356 C9VU5O 15462454 IC50 = 230 nM T78356 CLN4Z3 15462456 IC50 = 23 nM T78356 C1GSV2 15462460 IC50 = 25 nM T78356 CMU1C4 15462462 IC50 = 24.7 nM T78356 CV8Q6C 15586475 IC50 = 630 nM T78356 CBC0U6 15591372 IC50 = 10 nM T78356 CM1H0D 15684002 IC50 = 31.62 nM T78356 CPXY51 15684007 IC50 = 63.1 nM T78356 C7EA9P 15684009 IC50 = 50.12 nM T78356 C28YJT 15852309 IC50 = 3167 nM T78356 CK0V7J 15852311 IC50 = 82.1 nM T78356 C6I0DM 15852312 IC50 > 10000 nM T78356 C1WJ2D 16070041 IC50 = 3000 nM T78356 C5PO2I 18926535 IC50 = 34 nM T78356 CKIG56 18926585 IC50 = 19 nM T78356 C68KXJ 19003197 IC50 = 1100 nM T78356 C82UEL 19003218 IC50 = 850 nM T78356 C53TQI 19044744 IC50 = 10 nM T78356 CR12UN 19711412 IC50 = 47 nM T78356 C1SW6Y 22901615 IC50 = 1 nM T78356 CT84KG 23276768 IC50 = 6633 nM T78356 C43IRD 23276769 IC50 > 10000 nM T78356 C7CS3T 23276770 IC50 > 100000 nM T78356 CJ5CI8 23276771 IC50 = 2900 nM T78356 C4GJE1 23302977 IC50 = 38 nM T78356 C13JNA 23355384 IC50 = 940000 nM T78356 CS0X9N 23673433 IC50 = 7 nM T78356 CN59CD 24844985 IC50 = 200 nM T78356 C12JPW 24844986 IC50 = 100 nM T78356 CU6RA8 44209341 IC50 = 52 nM T78356 C7RS8L 44209342 IC50 = 24 nM T78356 CO53TB 44209343 IC50 = 51 nM T78356 C9RIT0 44209424 IC50 = 14 nM T78356 CC79FZ 44209484 IC50 = 19 nM T78356 CZE9V1 44209485 IC50 = 32 nM T78356 C3FWQ1 44209486 IC50 = 25 nM T78356 C3I0PU 44214442 IC50 = 640 nM T78356 CTC68R 44214443 IC50 = 1100 nM T78356 CLA5P3 44267574 IC50 = 85000 nM T78356 CFN56V 44267642 IC50 = 320000 nM T78356 C4DOG0 44269949 IC50 = 180 nM T78356 C59SXB 44269990 IC50 = 2100 nM T78356 CBXM82 44270004 IC50 = 4 nM T78356 CV28TF 44270371 IC50 = 18 nM T78356 C81VMD 44271591 IC50 = 900 nM T78356 CMF07P 44271601 IC50 = 4100 nM T78356 CZ78WQ 44271602 IC50 = 80 nM T78356 CGY72A 44271706 IC50 > 10000 nM T78356 C6S8KI 44271707 IC50 > 10000 nM T78356 C2GP6S 44271917 IC50 > 10000 nM T78356 C1BE2U 44271918 IC50 = 7400 nM T78356 C3O9JB 44272000 IC50 = 490 nM T78356 CSK27U 44272012 IC50 = 70 nM T78356 CL0GF6 44272014 IC50 = 50 nM T78356 CP5TK3 44277950 IC50 = 60 nM T78356 CX90IY 44278294 IC50 = 67 nM T78356 CHWG42 44278295 IC50 = 69 nM T78356 CM62IU 44278358 IC50 = 62 nM T78356 CL9N1T 44278387 IC50 > 10000 nM T78356 CT5OX9 44278388 IC50 > 5000 nM T78356 C3COK8 44278405 IC50 = 4200 nM T78356 CUO1T5 44278418 IC50 > 10000 nM T78356 CES49U 44278421 IC50 = 2900 nM T78356 CWH95I 44278426 IC50 > 10000 nM T78356 C7L5NH 44278442 IC50 = 960 nM T78356 CIW5V7 44278746 IC50 > 5000 nM T78356 C4JV6D 44278747 IC50 = 350 nM T78356 C9XDN8 44278750 IC50 > 10000 nM T78356 C5SIP8 44278834 IC50 = 6600 nM T78356 CK2A0N 44278856 IC50 = 1400 nM T78356 C8PH6W 44286986 IC50 = 770000 nM T78356 C2PI4C 44286987 IC50 = 1000000 nM T78356 C89IJC 44286988 IC50 = 470000 nM T78356 C5QZ3O 44286989 IC50 > 1000000 nM T78356 CP35AI 44287018 IC50 = 1000000 nM T78356 CZLR36 44287033 IC50 > 1000000 nM T78356 CR6B8Q 44287034 IC50 = 560000 nM T78356 CN2H8F 44287324 IC50 > 1000000 nM T78356 C46JGQ 44288679 IC50 = 26 nM T78356 C8Z9AU 44288680 IC50 = 43 nM T78356 CD6V9B 44288696 IC50 = 9 nM T78356 CI1BX5 44288697 IC50 = 7 nM T78356 CIWK56 44288859 IC50 = 3800 nM T78356 C61TCB 44288990 IC50 = 40 nM T78356 CP5T8Q 44289078 IC50 = 15 nM T78356 CJ2T4Z 44289086 IC50 = 80 nM T78356 C6C0EO 44289087 IC50 = 66 nM T78356 CS2D3R 44289090 IC50 = 43 nM T78356 CW46NZ 44289113 IC50 = 100 nM T78356 C95EHW 44289114 IC50 = 15 nM T78356 CNW35R 44289779 IC50 = 25 nM T78356 CA7JW1 44289893 IC50 = 71 nM T78356 CIO1W8 44292202 IC50 = 3300 nM T78356 CSUC58 44292203 IC50 = 19 nM T78356 CV1Q2E 44295569 IC50 = 29 nM T78356 C4S0NA 44295570 IC50 = 54 nM T78356 CQCH81 44295600 IC50 = 54 nM T78356 CTZ5R1 44295601 IC50 = 78 nM T78356 C0W7OU 44295894 IC50 > 2000 nM T78356 C9S5YD 44295905 IC50 = 7 nM T78356 CFX30I 44295911 IC50 = 50 nM T78356 CV8U7O 44295925 IC50 = 340 nM T78356 C5V2BJ 44295926 IC50 = 120 nM T78356 C7MF2H 44295945 IC50 = 790 nM T78356 C6BHK7 44295993 IC50 > 500 nM T78356 CD1VG9 44296070 IC50 = 125 nM T78356 C64XAN 44296071 IC50 = 165 nM T78356 CTU29Z 44297292 IC50 = 18 nM T78356 C69CMJ 44297354 IC50 = 4 nM T78356 C3B8ZY 44297392 IC50 = 20 nM T78356 CE4AX0 44297394 IC50 = 10 nM T78356 C7S5AC 44297768 IC50 = 2.3 nM T78356 C1JBN7 44301170 IC50 > 10000 nM T78356 CFR8S2 44301194 IC50 = 31.2 nM T78356 C13YUJ 44301318 IC50 = 82.1 nM T78356 CZ4GJ7 44305326 IC50 = 11 nM T78356 CS0YH6 44305343 IC50 = 10 nM T78356 C9O7JM 44305452 IC50 = 43 nM T78356 C4GLA1 44305478 IC50 > 200 nM T78356 C92WKH 44305481 IC50 > 100 nM T78356 CFQ9O3 44305522 IC50 = 17 nM T78356 CG2OL4 44305538 IC50 = 22 nM T78356 CB62ZJ 44305550 IC50 = 32 nM T78356 CT2CF5 44305675 IC50 > 200 nM T78356 CWZJ12 44305824 IC50 = 65 nM T78356 C0EC1W 44326402 IC50 > 10000 nM T78356 CP3ZE2 44326472 IC50 > 10000 nM T78356 C1X5NL 44326473 IC50 > 10000 nM T78356 CFIQ58 44326541 IC50 > 10000 nM T78356 CKA0O6 44326662 IC50 > 10000 nM T78356 C7GM2U 44326663 IC50 > 10000 nM T78356 CO2VC9 44330681 IC50 = 65 nM T78356 C6VU7R 44330682 IC50 = 75 nM T78356 CZYW38 44330686 IC50 = 29 nM T78356 CT1ZL9 44330902 IC50 = 55 nM T78356 CEM94D 44330919 IC50 = 63 nM T78356 C28JQI 44330921 IC50 = 250 nM T78356 CA5U6L 44330932 IC50 = 80 nM T78356 CSCT86 44330948 IC50 = 82 nM T78356 CVT09R 44330958 IC50 = 83 nM T78356 CQK19M 44330959 IC50 = 180 nM T78356 CI4WE7 44330972 IC50 = 41 nM T78356 C07WCL 44332831 IC50 = 78 nM T78356 CPL73O 44332843 IC50 = 22 nM T78356 CTS39I 44333045 IC50 = 15 nM T78356 CG53JD 44333064 IC50 = 39 nM T78356 CV0HK9 44333075 IC50 = 135 nM T78356 C4VY8X 44333097 IC50 = 20 nM T78356 C01LDO 44342814 IC50 = 88 nM T78356 CAU7P0 44342826 IC50 = 3.6 nM T78356 CG24OM 44343010 IC50 = 1.2 nM T78356 C54IEX 44343040 IC50 = 4.7 nM T78356 CL0T1C 44343042 IC50 = 12 nM T78356 CE7T6O 44343043 IC50 > 1000 nM T78356 C2YO6L 44343130 IC50 = 72 nM T78356 C7JC6O 44343184 IC50 = 44 nM T78356 CM6I9O 44343185 IC50 = 52 nM T78356 CX73JP 44343361 IC50 = 4.9 nM T78356 C01YFV 44343370 IC50 = 21 nM T78356 CB20SR 44343382 IC50 = 21 nM T78356 C9OVJ2 44343429 IC50 = 1.8 nM T78356 CW8XQ9 44350662 IC50 = 4 nM T78356 CYCS78 44350670 IC50 = 27 nM T78356 CQ1KR3 44353162 IC50 > 10000 nM T78356 CM60IB 44353169 IC50 = 39 nM T78356 CTI2M5 44353269 IC50 > 100000 nM T78356 C43AOM 44357779 IC50 = 90 nM T78356 C9CM5A 44357794 IC50 = 65 nM T78356 C64IWU 44358640 IC50 = 35000 nM T78356 C1XVD8 44366527 IC50 = 35.7 nM T78356 C1ASC2 44374425 IC50 = 40 nM T78356 CFG3R2 44374426 IC50 = 15 nM T78356 CLYA08 44374436 IC50 = 220 nM T78356 CU8K1E 44374438 IC50 = 42 nM T78356 CKW29G 44374442 IC50 = 90 nM T78356 C4ZO3W 44374443 IC50 = 50 nM T78356 CGKY24 44374452 IC50 = 44 nM T78356 C5KA6W 44374455 IC50 = 40 nM T78356 C54QJA 44374457 IC50 = 164 nM T78356 CVD81R 44374458 IC50 = 71 nM T78356 C6SP3M 44374462 IC50 = 500 nM T78356 C0LHQ3 44374492 IC50 = 20 nM T78356 C8LI5R 44374505 IC50 = 39 nM T78356 CU4N0J 44374506 IC50 = 46 nM T78356 CXPD94 44374507 IC50 = 280 nM T78356 C2H0XN 44374508 IC50 = 41 nM T78356 C09MVC 44374535 IC50 = 45 nM T78356 C6TDS3 44374545 IC50 = 45 nM T78356 C5Q9XG 44374548 IC50 = 45 nM T78356 CDG36Y 44374549 IC50 < 10 nM T78356 C4CG0B 44374558 IC50 < 10 nM T78356 C43AFG 44374559 IC50 = 37 nM T78356 CP4XW7 44374560 IC50 = 12 nM T78356 C3PB5V 44374590 IC50 = 40 nM T78356 CKZ8B7 44374623 IC50 = 40 nM T78356 CI15SX 44374634 IC50 = 40 nM T78356 CS6T4M 44374647 IC50 = 30 nM T78356 C0AYJ4 44374685 IC50 = 29 nM T78356 C1ZOS4 44374692 IC50 = 360 nM T78356 C2YT1N 44374696 IC50 = 42 nM T78356 C6ZQ3E 44374697 IC50 = 51 nM T78356 C0UOT1 44374698 IC50 = 34 nM T78356 C7BDM5 44374700 IC50 = 54 nM T78356 CR5LA6 44374701 IC50 = 48 nM T78356 CWU80E 44374721 IC50 = 39 nM T78356 C9I4ZT 44374740 IC50 = 37 nM T78356 CK1A0I 44374752 IC50 = 66 nM T78356 CAV4E2 44374837 IC50 = 199.53 nM T78356 CS9NZ5 44374845 IC50 = 31.62 nM T78356 CZ25PW 44374850 IC50 = 199.53 nM T78356 CQX8J7 44374857 IC50 = 39.81 nM T78356 CXY02H 44374860 IC50 = 199.53 nM T78356 CHT09F 44374886 IC50 < 1000 nM T78356 CHX8E3 44374895 IC50 = 50.12 nM T78356 C0WVL2 44374902 IC50 = 501.19 nM T78356 C4RQ6S 44374917 IC50 = 19.95 nM T78356 CO8Q1T 44374930 IC50 = 50 nM T78356 C07GQT 44374931 IC50 < 10 nM T78356 CT8EZ5 44374945 IC50 = 22 nM T78356 CMC19F 44374965 IC50 = 36 nM T78356 C7O3UE 44374966 IC50 = 60 nM T78356 C9MJA1 44374981 IC50 = 45 nM T78356 C79GUZ 44374982 IC50 = 26 nM T78356 CA61WC 44375026 IC50 = 79.43 nM T78356 CW82AO 44375168 IC50 = 50.12 nM T78356 CAYQ27 44377795 IC50 = 69 nM T78356 C3GZE7 44377810 IC50 > 1000 nM T78356 C7C3TH 44377817 IC50 = 465 nM T78356 CIAQ34 44377818 IC50 = 151 nM T78356 CQR0U2 44377819 IC50 = 24 nM T78356 CR0K6V 44377843 IC50 = 72 nM T78356 CT8D1J 44377844 IC50 = 68 nM T78356 C4WN9S 44377845 IC50 = 65 nM T78356 CG8F9I 44377846 IC50 = 58 nM T78356 CE3HO5 44377875 IC50 = 540 nM T78356 CCF7J8 44377882 IC50 > 1000 nM T78356 CZYU72 44377911 IC50 = 59 nM T78356 CV0H5A 44377912 IC50 = 80 nM T78356 C78KLA 44382602 IC50 = 50 nM T78356 C7CB6Q 44382605 IC50 = 9100 nM T78356 C2VJ3P 44382650 IC50 = 4600 nM T78356 CZ1K9H 44382651 IC50 = 1000 nM T78356 C0GP3M 44382653 IC50 = 3800 nM T78356 C6KF3P 44382656 IC50 = 1600 nM T78356 CC9IQ1 44382697 IC50 = 42 nM T78356 C4RQD7 44383249 IC50 = 9100 nM T78356 CF7IN2 44383250 IC50 = 24000 nM T78356 CF17HU 44383251 IC50 = 78000 nM T78356 CK56NY 44383252 IC50 = 44 nM T78356 C4OZ2M 44383253 IC50 = 2100 nM T78356 C0VWT5 44385499 IC50 = 400 nM T78356 C1A4GH 44385671 IC50 = 600 nM T78356 CS5TY4 44385778 IC50 = 300 nM T78356 CP9Y2Q 44385951 IC50 = 500 nM T78356 C37NWY 44386373 IC50 = 100 nM T78356 C60OVN 44386425 IC50 = 200 nM T78356 CG2XH3 44386636 IC50 = 40 nM T78356 CQHJ63 44387031 IC50 = 50 nM T78356 CI3BM4 44390722 IC50 = 1400 nM T78356 CF0YU5 44404186 IC50 = 78 nM T78356 CH1O6B 44457567 IC50 = 310 nM T78356 CRB3C5 44457587 IC50 = 5 nM T78356 C3XVR6 44458914 IC50 = 1020 nM T78356 CK4CU0 45259324 IC50 > 1000 nM T78356 C6GK7O 46213655 IC50 > 40000 nM T78356 CJP9O3 51346855 IC50 > 40000 nM T78356 C58DMR 53252516 IC50 > 50000 nM T78356 C08TYZ 53317604 IC50 > 40000 nM T78356 CN48MT 53326634 IC50 > 40000 nM T78356 C3IXM4 54728414 IC50 > 100000 nM T78356 C79DVG 56589615 IC50 > 3000 nM T78356 C9KGN4 70684971 IC50 = 230 nM T78356 CLMR38 71450832 IC50 > 10000 nM T78356 C6OQ3R 71451008 IC50 > 200 nM T78356 CEYX48 71454422 IC50 = 5.8 nM T78356 CI6B9U 71454429 IC50 = 4000 nM T78356 CXP2S8 71456310 IC50 > 200 nM T78356 C0FLT1 90655687 IC50 = 1000 nM T78356 D00RRV 792486 IC50 = 25 nM T78356 D01CGR 194468 IC50 = 15 nM T78356 D01IJX 10537337 IC50 = 5300 nM T78356 D01QOU 23663937 IC50 = 4.3 nM T78356 D01TOR 667555 IC50 = 5800 nM T78356 D04KDB 13885278 IC50 = 2000 nM T78356 D04ZGF 10561174 IC50 = 290 nM T78356 D05VAN 10331244 IC50 = 8.4 nM T78356 D09AUL 10266864 IC50 = 220 nM T78356 D09CPC 13728862 IC50 = 540 nM T78356 D0PU5V 10750911 IC50 = 5400 nM T78356 D0R8NE 13569172 IC50 = 660 nM T78356 D0TZ8C 14373279 IC50 = 380 nM T78356 D0U8YQ 921562 IC50 = 830 nM T78356 D0W6TB 16730275 IC50 = 30000 nM T78356 D0X8UK 10751574 IC50 = 1200 nM T78356 D0Y0QI 10774864 IC50 = 1500 nM T78356 D0Y1YZ 13569177 IC50 = 56 nM T82266 D00KHM 16362 IC50 = 162 nM T82266 D00STL 644241 IC50 = 4700 nM T82266 D01AXB 60835 IC50 = 2800 nM T82266 D01AZG 5073 IC50 = 34200 nM T82266 D01ZII 2726 IC50 = 3400 nM T82266 D02MLW 60753 IC50 = 62500 nM T82266 D03CJL 3168 IC50 = 7600 nM T82266 D03DAP 3356 IC50 = 27100 nM T82266 D03VPC 2754 IC50 = 91200 nM T82266 D04OSE 4485 Ki = 14.45 nM T82266 D04VMT 5253 IC50 = 193300 nM T82266 D04ZAH 43672 IC50 = 1226000 nM T82266 D06ABF 3957 IC50 = 11400 nM T82266 D06GDY 43815 IC50 = 3900 nM T82266 D06ZUK 3696 IC50 = 8300 nM T82266 D07ACT 5479530 IC50 = 153800 nM T82266 D07JVL 3016 IC50 = 30500 nM T82266 D07MVK 37393 IC50 = 1900 nM T82266 D07TQV 60825 IC50 = 54200 nM T82266 D07UYO 441401 IC50 = 105400 nM T82266 D09OJQ 4095 IC50 = 37400 nM T82266 D0A2ZX 4173 IC50 = 177900 nM T82266 D0B3UJ 115237 IC50 = 193900 nM T82266 D0CL9S 159269 IC50 = 713900 nM T82266 D0D1AL 3559 IC50 = 1700 nM T82266 D0E4DW 1775 IC50 = 21900 nM T82266 D0E6XR 3062316 IC50 = 81100 nM T82266 D0F0YZ 4737 IC50 = 299000 nM T82266 D0H3WI 37542 IC50 = 622500 nM T82266 D0I1FQ 54671008 IC50 = 246700 nM T82266 D0K6GZ 60464 IC50 = 88800 nM T82266 D0L4YD 154059 IC50 = 4300 nM T82266 D0L5WM 2157 IC50 = 270 nM T82266 D0M4YC 3114 IC50 = 1036700 nM T82266 D0N3VR 71616 IC50 = 414200 nM T82266 D0NS6H 3152 IC50 = 34300 nM T82266 D0NW3X 71329 IC50 = 26700 nM T82266 D0OB1J 39186 IC50 = 450 nM T82266 D0R0FE 2520 IC50 = 200 nM T82266 D0R0MW 5329102 IC50 = 33400 nM T82266 D0R3JB 4212 IC50 = 22500 nM T82266 D0S5CU 4499 IC50 = 0.015 nM T82266 D0U1OE 5452 IC50 = 3500 nM T82266 D0U2JP 4369359 IC50 = 147100 nM T82266 D0U5SI 4913 IC50 = 389500 nM T82266 D0WI3T 441243 IC50 = 1900 nM T82266 D0X0RI 4178 IC50 = 100000 nM T82266 D0Y4JJ 2351 IC50 = 1000 nM T82266 D0Y5UG 2160 IC50 = 11600 nM T82266 D0Z1RV 135398737 IC50 = 3600 nM T82266 D00ERV 1234 Ki = 5.4 nM T82266 D04TNT 46851313 IC50 > 10000 nM T82266 D0K9IF 71666749 IC50 > 30000 nM T82266 D0N1HW 5311200 IC50 = 9000 nM T82266 D0W8XT 60663 IC50 = 156 nM T82266 D0Y3ZP 23480 IC50 = 4800 nM T82266 D03SXN 104943 IC50 = 240 nM T82266 D08SOF 5405 IC50 = 930 nM T82266 D0OS6O 60149 IC50 = 6300 nM T82266 D0Y2HR 2247 IC50 = 1100 nM T82266 CPJ0C2 2747 IC50 = 30000 nM T82266 CZUI83 2769 IC50 = 11800 nM T82266 CGYS02 282663 IC50 = 0.046 nM T82266 CT15HN 341862 Ki = 32.8 nM T82266 CURH47 341863 Ki = 21.7 nM T82266 CLD6J9 441074 IC50 = 6400 nM T82266 CZYS12 501055 IC50 = 5300 nM T82266 C4R8TH 501058 IC50 > 10000 nM T82266 CP8ON7 501062 IC50 = 2700 nM T82266 C5QLA6 9827668 IC50 = 2300 nM T82266 CQ4LC2 9872676 Ki = 145 nM T82266 CVJ7I8 9910573 IC50 = 1526 nM T82266 CPBQ94 9948049 IC50 = 2700 nM T82266 C5K6MJ 9976640 IC50 = 980 nM T82266 CNJA83 10091655 IC50 = 0.0081 nM T82266 CYXB38 10414981 IC50 > 10000 nM T82266 CWL1K9 10874724 IC50 = 4840 nM T82266 CRI50E 10885636 IC50 = 1720 nM T82266 CX65PW 10907460 IC50 = 860 nM T82266 CSLT97 10949380 IC50 = 1710 nM T82266 CJC9K4 11005810 IC50 = 284 nM T82266 C56YON 11069321 IC50 = 308 nM T82266 CG41BK 11071079 IC50 = 2730 nM T82266 C7DE0U 11113605 IC50 = 4300 nM T82266 CU6PV0 11143820 IC50 = 1110 nM T82266 C7PVL8 11730467 IC50 = 2350 nM T82266 CN9M8E 11811722 IC50 = 552 nM T82266 C5XJP9 13069167 IC50 = 0.045 nM T82266 CNJW02 13069170 IC50 = 0.033 nM T82266 CK8V5X 13069171 IC50 = 0.03 nM T82266 CNEM42 13121206 IC50 = 0.05 nM T82266 CK6N9E 13181322 Ki = 29.9 nM T82266 CJ6X5E 13233216 IC50 = 0.01 nM T82266 COZ8Q5 13912577 IC50 = 5.2 nM T82266 C18BOL 13912583 IC50 = 710 nM T82266 CL1HD9 13934401 IC50 = 140 nM T82266 CZ1O3S 13957269 IC50 = 160 nM T82266 CA06UQ 14788031 IC50 = 17 nM T82266 CZ8WK5 14788032 IC50 = 3.1 nM T82266 CE36FM 14788033 IC50 = 88 nM T82266 C3VM1R 14788034 IC50 = 17 nM T82266 C0IZA1 14788035 IC50 = 280 nM T82266 CNCB03 14788036 IC50 = 26 nM T82266 C3JD9A 14788037 IC50 = 1.5 nM T82266 C8BLX9 14788038 IC50 = 2.7 nM T82266 C5VZY4 14788039 IC50 = 100 nM T82266 CFWR73 14788040 IC50 = 1.7 nM T82266 CPMT85 14788041 IC50 = 2 nM T82266 C9MXA0 14788042 IC50 = 1500 nM T82266 CC9UY7 14788043 IC50 = 3.6 nM T82266 C8G6RF 14788044 IC50 = 14 nM T82266 CB35GD 14788045 IC50 = 11 nM T82266 CCZ3Y6 14788046 IC50 = 270 nM T82266 CT7WQ5 14788047 IC50 = 50 nM T82266 CHT2Q0 14788049 IC50 = 2.6 nM T82266 CB64EN 16049818 IC50 = 20000 nM T82266 CFQM24 20664161 IC50 > 10000 nM T82266 C0LR3P 22859115 IC50 = 580 nM T82266 C8T7NC 25118805 IC50 > 10000 nM T82266 CCZ07E 44283398 IC50 = 0.39 nM T82266 CBXD38 44283427 IC50 = 0.017 nM T82266 CNY68K 44283656 IC50 = 0.022 nM T82266 CQIZ12 44284652 IC50 = 26 nM T82266 C3W9ZL 44284918 IC50 = 4 nM T82266 C1A5CW 44299271 IC50 = 1670 nM T82266 C9R7BI 44299273 IC50 = 5500 nM T82266 C3WP5N 44326361 IC50 > 10000 nM T82266 C6LM8X 44334364 IC50 = 0.14 nM T82266 C56TLX 44334371 IC50 = 0.25 nM T82266 CMI83R 44334376 IC50 = 2.8 nM T82266 CBU80L 44334381 IC50 = 0.013 nM T82266 C9X1VK 44334386 IC50 = 1.5 nM T82266 C58ZUX 44334389 IC50 = 0.027 nM T82266 CZW93T 44334390 IC50 = 2.3 nM T82266 CD9ZS8 44342270 IC50 = 1340 nM T82266 CATD12 44401751 IC50 > 10000 nM T82266 C16MBG 44401760 IC50 > 10000 nM T82266 CPWV46 44550725 IC50 = 14070 nM T82266 C73XBL 57384077 IC50 = 1900 nM T82266 CV2T7S 70691408 IC50 = 71000 nM T82266 CFMJ96 119081417 IC50 = 3000 nM T82266 COK4D6 135401985 IC50 > 30000 nM T82266 C1DM3K 135401987 IC50 > 30000 nM T82266 CC16GW 137625280 IC50 = 26000 nM T82266 CIY0P1 137632867 IC50 = 90080 nM T82266 CH05QS 137633237 IC50 > 10000 nM T82266 C8IM4P 137637833 Ki = 36 nM T82266 C4YD3A 137639105 IC50 > 10000 nM T82266 CE41MQ 137641298 IC50 = 208 nM T82266 CM8LO4 137643183 IC50 = 127 nM T82266 CS87DF 137645885 IC50 > 10000 nM T82266 C1VQO6 137645918 IC50 = 516 nM T82266 C3JE5U 137652980 IC50 = 3766 nM T82266 C38FXZ 137653443 IC50 > 80000 nM T82266 CD1L5S 137657500 IC50 = 2706 nM T82266 COXF43 137658445 IC50 = 603 nM T82266 CUJ58E 137658891 IC50 = 909 nM T82266 CL2OR1 145950976 IC50 > 80000 nM T82266 CWPH76 155512737 IC50 = 4000 nM T82266 CTR7C8 155516568 IC50 = 25000 nM T82266 CWD04K 155525738 IC50 = 2800 nM T82266 CZ10BI 155536168 IC50 = 16000 nM T82266 CT6UN1 155541545 IC50 = 24000 nM T82266 CNQ0F4 155544914 IC50 = 15000 nM T82266 CQE7F8 155548011 IC50 = 1500 nM T82266 CZ8W0Y 155551407 IC50 = 2900 nM T82266 CJQ59S 155563181 IC50 = 21000 nM T82266 D01BWV 9802572 IC50 = 128 nM T82266 D0U7OD 16043230 IC50 = 730 nM T36557 D00WCX 39042 EC50 = 18900 nM T36557 D0G2MW 446284 IC50 = 4000 nM T36557 D0N6RF 65999 EC50 > 10000 nM T36557 D0NF1U 64929 EC50 > 10000 nM T36557 D0O1TC 5280581 IC50 = 4300 nM T36557 D0UE9X 5280933 IC50 = 750 nM T36557 D03OSG 11236126 EC50 = 1.9 nM T36557 D04BPS 9888484 IC50 = 1914.26 nM T36557 D04QIE 11526038 EC50 = 1580 nM T36557 D0I5IM 135449333 IC50 = 3800 nM T36557 D0LW1Y 9864881 EC50 = 10 nM T36557 D0M0SS 170364 Ki = 1200 nM T36557 D0U0KR 3035850 Ki = 0.43 nM T36557 D0H5FI 9958543 IC50 > 15000 nM T36557 D05HDX 9803963 Ki = 0.048 nM T36557 D08LZI 9947731 EC50 > 100000 nM T36557 D0B0EB 9890585 IC50 = 5248.07 nM T36557 D0B8JQ 9825046 EC50 = 1920 nM T36557 D0B9EN 10274777 EC50 = 53 nM T36557 C9RN3W 7127 EC50 = 50600 nM T36557 CSB8Q0 8215 IC50 = 30000 nM T36557 CVT2C4 10467 IC50 = 30000 nM T36557 C35BMO 82145 EC50 = 3720 nM T36557 CB5H9D 89954 EC50 > 100000 nM T36557 C69SGI 312225 EC50 = 112 nM T36557 CUC68S 339720 EC50 = 230 nM T36557 C1PJ5Z 443023 EC50 = 18110 nM T36557 C12SCN 637584 EC50 = 49500 nM T36557 CZN6S9 743974 IC50 > 25118.86 nM T36557 C9KP6J 1285388 IC50 = 34000 nM T36557 CAQI34 3033829 EC50 > 100000 nM T36557 CT29VZ 4388708 EC50 = 21000 nM T36557 C32LKN 4518233 IC50 = 389941.99 nM T36557 CH34WN 5281116 IC50 = 30000 nM T36557 C6K2GJ 5281805 EC50 = 22340 nM T36557 C75ORQ 5310669 EC50 = 24390 nM T36557 CZ0D2P 5715241 EC50 = 12440 nM T36557 CZJ84H 6102812 IC50 = 223 nM T36557 C16ZSG 6439929 EC50 > 100000 nM T36557 CI2GA0 6992117 EC50 > 100000 nM T36557 CGXH64 9547900 EC50 = 10 nM T36557 C50PDQ 9549255 EC50 = 70 nM T36557 C5PGB8 9803821 EC50 = 6000 nM T36557 CQK19U 9822766 EC50 = 700 nM T36557 C47ZRD 9823501 EC50 = 90 nM T36557 CSY86D 9825523 IC50 = 490 nM T36557 CJF2M6 9826186 IC50 = 1900 nM T36557 CR7J1B 9844286 IC50 = 340 nM T36557 CSZ36U 9844554 EC50 = 3310 nM T36557 C0Z2DQ 9845736 EC50 = 3000 nM T36557 C9RM5A 9845832 EC50 = 30 nM T36557 C6ABL9 9850395 EC50 = 5000 nM T36557 C7S3YF 9866595 Ki = 2500 nM T36557 CWJU60 9870703 EC50 = 100 nM T36557 C5GA7U 9888528 EC50 = 1500 nM T36557 CED08V 9889284 EC50 = 315 nM T36557 C6O1SV 9895808 EC50 = 19 nM T36557 C62YXO 9910188 EC50 = 2.1 nM T36557 C1G6FX 9932058 EC50 = 420 nM T36557 C75NOF 9932563 EC50 = 20 nM T36557 C9PCJ5 9932790 EC50 = 10 nM T36557 CGV83S 9933541 EC50 = 3000 nM T36557 CF7P8W 9934050 IC50 = 170 nM T36557 CPUF90 9952559 EC50 = 2800 nM T36557 CPMH16 9953945 EC50 = 30 nM T36557 C2VHT3 9955922 IC50 > 15000 nM T36557 CRE2W1 9956726 EC50 = 2600 nM T36557 CQP9I8 9960726 EC50 = 10500 nM T36557 CJA73Y 9980571 EC50 = 5 nM T36557 CV74OZ 9980586 EC50 = 2400 nM T36557 C45OEJ 9980930 IC50 = 834 nM T36557 CFKD10 9981617 IC50 > 15000 nM T36557 C27AED 9982759 EC50 = 3.4 nM T36557 CH7W9P 10003213 EC50 = 2.9 nM T36557 CKJ83Z 10004270 IC50 = 5519 nM T36557 C8JV7T 10004390 Ki = 93 nM T36557 CUE80O 10004438 EC50 = 1.9 nM T36557 CIZJ14 10005136 IC50 > 15000 nM T36557 C6VP7J 10005230 IC50 > 15000 nM T36557 CK24FM 10005763 EC50 = 5.2 nM T36557 C0OED7 10023279 EC50 > 10000 nM T36557 C45ZDO 10026148 EC50 = 3 nM T36557 C0RVG2 10027920 EC50 = 58 nM T36557 C7H4RX 10050194 EC50 = 9 nM T36557 CQH15A 10053715 EC50 = 53 nM T36557 C48JGT 10070650 EC50 = 6500 nM T36557 CNS96V 10072967 EC50 > 10000 nM T36557 CJRY94 10074505 EC50 = 3.4 nM T36557 CC72JH 10074964 EC50 = 18 nM T36557 C79TZB 10075037 EC50 = 46 nM T36557 CO2IN7 10075041 EC50 = 3.2 nM T36557 C9PH1M 10075336 EC50 = 3.3 nM T36557 CM5EU7 10093355 EC50 = 9550 nM T36557 C3ZT0K 10096907 IC50 = 372 nM T36557 CQ2EH0 10096908 IC50 = 892 nM T36557 CRJU50 10098103 EC50 = 320 nM T36557 CZU39A 10113515 IC50 = 4123 nM T36557 CW5KR2 10113686 IC50 > 15000 nM T36557 CQG9E4 10113721 EC50 = 120 nM T36557 CWH2U3 10113980 IC50 = 740 nM T36557 C1BA8V 10114442 IC50 = 10495.42 nM T36557 C6FIV9 10115344 IC50 = 1569 nM T36557 C1EOY3 10116365 IC50 > 50000 nM T36557 C15GVJ 10116451 IC50 > 15000 nM T36557 CY73BR 10117908 EC50 = 830 nM T36557 CTGB91 10118056 IC50 > 50000 nM T36557 CRCG14 10118927 Ki = 7 nM T36557 C74VJE 10136660 IC50 = 3935.5 nM T36557 CDX37J 10137693 IC50 = 7600 nM T36557 CVI26N 10138146 EC50 > 10000 nM T36557 CMRP39 10139247 IC50 = 7112.14 nM T36557 C6RPI1 10139836 IC50 > 50000 nM T36557 C6N1TJ 10140233 IC50 > 50000 nM T36557 CR4E1D 10141305 EC50 > 10000 nM T36557 CB53WS 10141607 EC50 = 678 nM T36557 C7XT5K 10159635 EC50 > 10000 nM T36557 CCT52G 10160395 EC50 = 1.1 nM T36557 C9C3JQ 10162008 IC50 = 1698.24 nM T36557 CZ24HT 10162063 EC50 > 10000 nM T36557 C7DU6F 10162210 IC50 > 15000 nM T36557 CDM26O 10162519 IC50 > 15000 nM T36557 CMF69H 10162615 IC50 > 50000 nM T36557 C6AE1Y 10163556 EC50 > 10000 nM T36557 C9FR3O 10174350 EC50 = 13 nM T36557 CDT75W 10182946 IC50 > 15000 nM T36557 C7I1LS 10183245 IC50 = 1250 nM T36557 CUQ89L 10183490 IC50 = 1999.86 nM T36557 C49HSN 10183977 IC50 > 50000 nM T36557 C89CVS 10186123 EC50 = 520 nM T36557 CPM13H 10201545 EC50 = 120 nM T36557 CC3G0I 10204762 IC50 = 2300 nM T36557 CAQ5U8 10205828 IC50 > 50000 nM T36557 CMSG62 10207241 IC50 > 15000 nM T36557 C6MYJ4 10207242 IC50 > 50000 nM T36557 CM4HS7 10207244 IC50 > 50000 nM T36557 C27EYG 10207287 EC50 = 1100 nM T36557 C30RKL 10207974 EC50 = 5900 nM T36557 CO52SH 10208214 IC50 > 50000 nM T36557 C1NIA4 10217191 IC50 = 3.1 nM T36557 CL1K2N 10223023 IC50 = 1389.95 nM T36557 CY28GC 10224783 IC50 > 15000 nM T36557 CQ56VG 10225637 IC50 > 50000 nM T36557 CJH81C 10225731 IC50 > 50000 nM T36557 CYR3B5 10226233 IC50 = 2322.74 nM T36557 CG4P7X 10226511 IC50 = 6900 nM T36557 CSL75P 10228304 IC50 = 4220 nM T36557 CS7Q9U 10229225 IC50 > 50000 nM T36557 CY38EO 10230466 EC50 = 2300 nM T36557 COVB68 10252612 EC50 = 4600 nM T36557 CC8GU0 10254028 EC50 = 2.5 nM T36557 CARH74 10254209 EC50 = 1700 nM T36557 C2HIT7 10254845 IC50 = 259 nM T36557 C4PM2S 10274627 EC50 = 4 nM T36557 CZ64AI 10275334 EC50 = 5400 nM T36557 CI1BV7 10276470 IC50 > 15000 nM T36557 C7YMO1 10276539 IC50 = 5137 nM T36557 CIOK04 10277666 IC50 > 15000 nM T36557 C02EHS 10279905 IC50 > 15000 nM T36557 CW34DF 10280116 EC50 = 8240 nM T36557 CSJ28C 10280496 IC50 > 15000 nM T36557 CS1U0K 10281422 IC50 > 50000 nM T36557 CQR18V 10295993 EC50 > 10000 nM T36557 CK7F1O 10297427 IC50 > 50000 nM T36557 CO1P5R 10297760 IC50 = 7498.94 nM T36557 CL40QG 10297943 EC50 > 10000 nM T36557 CL5WB3 10299983 IC50 > 50000 nM T36557 CS9V4N 10300072 IC50 > 50000 nM T36557 C89QXN 10300073 IC50 > 50000 nM T36557 C7UNX1 10300279 EC50 = 4600 nM T36557 CLQD46 10301814 IC50 > 50000 nM T36557 CFS25Z 10320822 EC50 = 2400 nM T36557 CQH6P7 10323352 EC50 = 3.5 nM T36557 CDU6H7 10323599 EC50 = 3 nM T36557 CGD4N7 10341169 EC50 = 8400 nM T36557 C01MTP 10341401 EC50 = 1270 nM T36557 C6HM5O 10342769 EC50 = 2500 nM T36557 C8AT6R 10342801 IC50 > 15000 nM T36557 C3NJ4S 10343538 EC50 = 2500 nM T36557 CB6R4D 10344769 EC50 = 1400 nM T36557 CPT82D 10347115 EC50 = 4.4 nM T36557 C23JXU 10367018 IC50 > 15000 nM T36557 C84KIW 10367602 EC50 = 34 nM T36557 C0SKH9 10368050 IC50 = 5230 nM T36557 CMW4U5 10368444 EC50 = 3.3 nM T36557 CC1IK3 10370262 EC50 = 17 nM T36557 C0SLF7 10371709 EC50 = 2170 nM T36557 CN92GI 10387634 EC50 = 7900 nM T36557 CLI13C 10390756 EC50 = 28 nM T36557 C4GD0W 10408561 EC50 = 2450 nM T36557 CQY70C 10409988 EC50 > 10000 nM T36557 C9GLW7 10410878 EC50 = 5000 nM T36557 CJB86G 10411897 EC50 = 10 nM T36557 C29PFI 10412116 EC50 = 2400 nM T36557 C72JHZ 10432356 EC50 > 10000 nM T36557 CEO2U1 10432525 EC50 = 900 nM T36557 CTQ0R7 10433053 EC50 > 10000 nM T36557 CKGE28 10434749 EC50 = 218 nM T36557 C63QBA 10455509 EC50 = 2400 nM T36557 CWQ2K1 10455511 EC50 = 2500 nM T36557 CT7PM6 10455681 EC50 = 1.6 nM T36557 C1S7GU 10455871 EC50 = 1.3 nM T36557 C4DXE1 10457843 EC50 = 4.1 nM T36557 C1H5RP 10458842 EC50 = 1.9 nM T36557 C9Q5HV 10480558 EC50 = 6000 nM T36557 CJ6S2A 10480923 EC50 = 2 nM T36557 CP04MX 10481007 EC50 = 6 nM T36557 C8KNR9 10743135 EC50 = 790 nM T36557 CZG96J 10896097 EC50 = 29300 nM T36557 C5J4PX 10896495 EC50 = 23100 nM T36557 C9PIM1 10916251 EC50 = 8000 nM T36557 CJBM20 11042473 EC50 = 22600 nM T36557 CF38JZ 11048469 EC50 = 3000 nM T36557 CG23SM 11071056 EC50 = 15600 nM T36557 CV7UL0 11090513 EC50 = 640 nM T36557 CZD8U3 11101345 EC50 = 400 nM T36557 CR26YH 11111473 EC50 = 6600 nM T36557 C61TQH 11154732 EC50 = 46.7 nM T36557 CQ13LJ 11155087 IC50 = 2.999 nM T36557 CG2V4U 11155122 EC50 = 25 nM T36557 CIV54T 11155356 EC50 = 4.6 nM T36557 C3LG4F 11155783 EC50 = 1060 nM T36557 CN7QF3 11166818 EC50 = 1360 nM T36557 CIW98T 11167613 EC50 = 1550 nM T36557 CF0H2Q 11167738 EC50 > 25000 nM T36557 C3OWD7 11169884 EC50 = 2080 nM T36557 C4W7XI 11178006 IC50 = 2.999 nM T36557 CW2FH7 11178750 IC50 = 9682.78 nM T36557 CM3BO2 11178916 IC50 = 5074 nM T36557 C6BQ7O 11179502 EC50 > 25000 nM T36557 CK84AR 11188766 IC50 = 7.7 nM T36557 C2D9FS 11190667 EC50 = 1630 nM T36557 CA7K4Q 11190685 EC50 = 15.2 nM T36557 C7B0QN 11190733 IC50 > 50000 nM T36557 C89UCH 11202658 IC50 > 50000 nM T36557 C2JK4F 11203145 EC50 > 10000 nM T36557 CYHZ54 11208735 EC50 = 17170 nM T36557 C7ZPE1 11211156 EC50 = 65.5 nM T36557 C7P2LF 11214000 EC50 > 10000 nM T36557 C3G7FR 11214539 EC50 = 3 nM T36557 C8JZ6Q 11225048 EC50 = 2060 nM T36557 C8ATL5 11225797 EC50 = 370 nM T36557 CJ78RY 11225851 EC50 = 13 nM T36557 CE4I3N 11225910 EC50 = 60 nM T36557 CD2NX7 11227195 EC50 > 25000 nM T36557 C7ROX3 11235560 IC50 = 5 nM T36557 CK4F7Q 11235859 EC50 = 5 nM T36557 CQ3C1F 11235892 EC50 = 18 nM T36557 C2IBK8 11236542 IC50 > 50000 nM T36557 CBU98W 11236923 EC50 = 1600 nM T36557 CF31OJ 11237218 EC50 = 35 nM T36557 CGAI13 11237761 IC50 > 50000 nM T36557 CG8IQ1 11246863 EC50 = 26.8 nM T36557 CP1X0G 11247654 IC50 = 2 nM T36557 C7C9MZ 11247664 EC50 = 10 nM T36557 CBS49N 11247908 EC50 > 25000 nM T36557 C5VB4A 11248512 IC50 > 15000 nM T36557 C79VCR 11249385 IC50 = 5000 nM T36557 C7LK0I 11258987 EC50 = 2620 nM T36557 CJ6ON0 11259787 EC50 > 25000 nM T36557 CH9X1P 11260214 EC50 = 2100 nM T36557 C9J3DR 11271060 IC50 = 4448 nM T36557 C7ZC0P 11271211 EC50 = 2870 nM T36557 CYD12Z 11271514 EC50 = 2700 nM T36557 CWH02S 11280270 EC50 = 216 nM T36557 CH69MT 11281802 EC50 = 93 nM T36557 CH0K3Y 11282309 EC50 = 69.6 nM T36557 CNG61K 11282914 IC50 > 50000 nM T36557 C2O3WX 11283113 EC50 > 25000 nM T36557 CP0H1J 11293283 EC50 > 1000 nM T36557 CDK79P 11293459 EC50 = 237 nM T36557 CDX50Z 11293589 EC50 = 22.3 nM T36557 C6T9OR 11294565 EC50 = 5600 nM T36557 C5S6YO 11294660 EC50 = 7740 nM T36557 CFTW52 11295349 EC50 = 4 nM T36557 CMC6I8 11305717 EC50 = 7 nM T36557 CC81HS 11306364 EC50 = 5290 nM T36557 CDKC74 11306495 EC50 > 1000 nM T36557 C2KZ3M 11306745 EC50 > 25000 nM T36557 CG2D3O 11316534 EC50 = 35.4 nM T36557 CB12CE 11316788 EC50 = 70 nM T36557 C7Z1NC 11317347 EC50 = 102 nM T36557 CHO5P0 11327951 IC50 = 11 nM T36557 C1OEB0 11328910 EC50 = 33 nM T36557 C9SB2M 11329011 EC50 = 610 nM T36557 CIAP50 11329280 EC50 = 52 nM T36557 CSF2L4 11329304 EC50 = 1150 nM T36557 CRM6D3 11339310 EC50 = 23.3 nM T36557 CMCD29 11339649 IC50 > 15000 nM T36557 C6WI0Z 11339975 IC50 = 4100 nM T36557 C9B0LH 11340275 EC50 > 1000 nM T36557 CG91XM 11340322 EC50 = 26 nM T36557 C0ABC9 11340513 EC50 = 45 nM T36557 CLFX14 11340991 IC50 = 7232 nM T36557 C0LU6S 11349723 EC50 = 238 nM T36557 CQ7OF6 11351221 EC50 = 6.9 nM T36557 CEZG39 11351266 EC50 = 25 nM T36557 C72GEN 11351550 EC50 = 93 nM T36557 CL7D8V 11351980 IC50 > 15000 nM T36557 C9PAJ6 11352187 EC50 = 58 nM T36557 C7W1FO 11352276 EC50 = 45.5 nM T36557 CQN0X9 11352573 EC50 = 38 nM T36557 CET87Y 11352791 EC50 > 25000 nM T36557 C8VT0Y 11362757 EC50 = 3000 nM T36557 CM7TX9 11363175 IC50 > 50000 nM T36557 C6A3OW 11373952 EC50 = 147 nM T36557 CXHU81 11374318 EC50 = 10000 nM T36557 CKE9R8 11374679 EC50 > 10000 nM T36557 CDQ2M5 11374680 EC50 = 2165 nM T36557 CJI2C6 11376123 EC50 = 25000 nM T36557 C5TZY0 11385663 IC50 = 1190 nM T36557 C3Z1LN 11386159 EC50 = 3 nM T36557 C8WVM5 11386220 IC50 > 50000 nM T36557 C5OB8J 11386857 EC50 > 10000 nM T36557 C8X5PW 11393977 EC50 = 6400 nM T36557 C6SYD8 11396352 EC50 > 500 nM T36557 CTU8G6 11397018 EC50 = 2000 nM T36557 C0TX7O 11397203 EC50 = 12 nM T36557 CQ5CZ2 11397569 EC50 = 8.6 nM T36557 CXIN63 11397705 EC50 = 1700 nM T36557 COK68W 11399560 EC50 = 1800 nM T36557 CGY28A 11405204 EC50 = 711 nM T36557 CZB52S 11408244 EC50 > 10000 nM T36557 C34QBC 11408475 IC50 = 2685 nM T36557 CX7W4S 11408502 IC50 > 15000 nM T36557 CPB8F6 11409173 IC50 = 3 nM T36557 CCAJ14 11418941 EC50 = 0.06 nM T36557 C6Q8FR 11419459 EC50 = 2700 nM T36557 CMT65A 11421645 EC50 = 23.9 nM T36557 CCD7X1 11421714 EC50 = 2747 nM T36557 CZ3VT9 11430761 IC50 > 50000 nM T36557 C60KVM 11431103 EC50 = 1 nM T36557 C5SKD2 11431192 IC50 = 6745.28 nM T36557 CPGX09 11431289 EC50 = 6 nM T36557 C1OZ5D 11431625 EC50 = 2 nM T36557 CFU62G 11432162 EC50 = 2050 nM T36557 C6FP3T 11441763 EC50 = 54.3 nM T36557 CT4NR0 11442228 EC50 > 500 nM T36557 C2ZVF9 11442294 EC50 = 4850 nM T36557 CV5M3A 11442379 EC50 = 114 nM T36557 C4ZE1C 11465146 EC50 = 3 nM T36557 C6G7FO 11475460 EC50 = 49.8 nM T36557 CN64KX 11475461 EC50 = 138 nM T36557 C7ZO8B 11476297 EC50 = 3.4 nM T36557 CLZ5I1 11476382 IC50 > 15000 nM T36557 CI8FO6 11476916 EC50 = 8 nM T36557 CSX3Z0 11477433 EC50 > 25000 nM T36557 C83GWX 11477735 EC50 > 1000 nM T36557 CQ6L9S 11486733 EC50 = 17.1 nM T36557 C4S6JR 11488006 EC50 = 2.1 nM T36557 CZ84QA 11488726 IC50 = 3 nM T36557 C6HO8J 11490050 EC50 = 17 nM T36557 CL2V9K 11497604 EC50 = 80 nM T36557 CF1AI0 11503439 EC50 > 4200 nM T36557 CU27FT 11503588 EC50 = 125 nM T36557 C0JEO8 11511317 EC50 > 10000 nM T36557 C68RSH 11525752 IC50 = 69.98 nM T36557 CH14EK 11526493 IC50 = 5377 nM T36557 CT9Z0X 11539510 EC50 > 6300 nM T36557 C6IO2H 11547473 EC50 = 3 nM T36557 C5H7FP 11563028 IC50 > 50000 nM T36557 CF2V1D 11583815 IC50 = 2568 nM T36557 C3GI8R 11585006 EC50 = 7 nM T36557 C1HG4A 11591164 IC50 > 50000 nM T36557 CC15AQ 11592357 IC50 > 50000 nM T36557 C2ZP9O 11612623 EC50 = 80 nM T36557 CE87MQ 11619439 EC50 = 3000 nM T36557 C5LVA3 11620018 EC50 = 320 nM T36557 C4M5SU 11620299 EC50 = 0.9 nM T36557 CWOD63 11620575 IC50 > 50000 nM T36557 CQN62W 11626766 IC50 = 24 nM T36557 CR30AV 11627288 EC50 = 610 nM T36557 C4ZR8D 11627859 EC50 = 627 nM T36557 CM6R1L 11640895 EC50 = 4350 nM T36557 C89TBG 11649750 EC50 = 11 nM T36557 C16CWN 11649783 EC50 = 10 nM T36557 CTW7E6 11655554 IC50 = 1800 nM T36557 CY2DE9 11656305 EC50 = 9170 nM T36557 CD0NU7 11663038 EC50 = 3340 nM T36557 CL7C1Z 11663931 EC50 = 12 nM T36557 CQ2M8V 11669781 IC50 = 57.02 nM T36557 C27FGM 11677450 EC50 = 80 nM T36557 CHA36Y 11678044 IC50 = 2398.83 nM T36557 C6H8PJ 11678481 EC50 = 14 nM T36557 C8MU1C 11683336 EC50 = 23 nM T36557 CD43TA 11698802 IC50 > 50000 nM T36557 C3FIK4 11704026 EC50 = 7900 nM T36557 CGK13J 11705301 IC50 = 79 nM T36557 CR46YH 11705832 EC50 = 4000 nM T36557 C2WQ1O 11711595 EC50 = 12 nM T36557 C5AX8M 11712774 EC50 = 2130 nM T36557 C2UY7P 11712873 EC50 = 243 nM T36557 C6C9HF 11741962 IC50 = 3500 nM T36557 CNQ6O1 11750720 EC50 = 28.4 nM T36557 CR7Y2E 11751021 IC50 = 3 nM T36557 C1ZR9N 11751796 EC50 = 45.6 nM T36557 C0Q4XH 11753952 Ki = 0.3 nM T36557 C35DKP 11754345 EC50 = 4 nM T36557 CLE5P8 11754583 IC50 > 15000 nM T36557 C7O6FH 11755396 EC50 = 3.4 nM T36557 C18XBA 11755655 IC50 = 399 nM T36557 CL4EK8 11755968 EC50 = 11 nM T36557 CBV25C 11774828 EC50 = 6 nM T36557 CE27GQ 11775099 IC50 = 7040 nM T36557 C3EXH7 11775225 EC50 > 10000 nM T36557 CX5YP8 11784860 EC50 > 25000 nM T36557 CW8R9F 11785036 EC50 = 5 nM T36557 CZ52VY 11813713 Ki = 0.16 nM T36557 CL7V4Z 11826628 EC50 = 3100 nM T36557 C38KZG 11978565 EC50 > 100000 nM T36557 COPI61 11997929 EC50 = 2.6 nM T36557 C0XE9L 12870589 EC50 > 1000 nM T36557 CWL9C6 12967684 EC50 = 3000 nM T36557 CS82RI 14427412 EC50 = 4900 nM T36557 C0LH2E 15942850 EC50 = 500 nM T36557 CF6I7X 15981441 EC50 = 977 nM T36557 CDFT16 15984029 EC50 = 500 nM T36557 CEL3S6 16007090 EC50 = 15 nM T36557 C9T1QR 16036021 EC50 > 10000 nM T36557 CT3VA7 16036134 EC50 > 10000 nM T36557 CO5B2T 16043249 EC50 = 10 nM T36557 CY13OS 16046718 EC50 = 2000 nM T36557 CPY13K 16046721 EC50 = 2000 nM T36557 CTP15X 16046722 EC50 > 10000 nM T36557 C7AIM9 16048150 EC50 = 441 nM T36557 CY09JO 16048652 EC50 = 1.5 nM T36557 C5V0ZY 16085979 EC50 = 339 nM T36557 CD3K9X 16085980 EC50 = 5 nM T36557 CY1Q3Z 16085981 EC50 = 2 nM T36557 C1F6CM 16085982 IC50 = 5 nM T36557 C97HJA 16085983 IC50 = 5.998 nM T36557 CE3HN1 16085984 EC50 = 25 nM T36557 C2F4AJ 16085985 IC50 = 3.999 nM T36557 CE4Q7N 16085986 EC50 = 1 nM T36557 CXYF29 16085987 EC50 = 34 nM T36557 CPQ2K9 16085988 EC50 = 6 nM T36557 CF4J1K 16090330 EC50 = 1320 nM T36557 CU63PB 16090857 EC50 > 10000 nM T36557 CA51QP 16090858 EC50 = 4300 nM T36557 C8O1HI 16090859 EC50 = 4630 nM T36557 CMKI28 16090878 EC50 = 6980 nM T36557 CJC53L 16090879 EC50 > 10000 nM T36557 CJ3D4H 16109183 EC50 = 20 nM T36557 CJ38DY 16109187 EC50 > 10000 nM T36557 CS8NF6 16109190 EC50 = 4050 nM T36557 C9IO5Z 16109193 EC50 > 25000 nM T36557 CU0BK1 16109199 EC50 = 6260 nM T36557 C2S0TO 16109209 EC50 = 808 nM T36557 C7V9EL 16109210 EC50 > 10000 nM T36557 CP0SB8 16110418 EC50 = 44 nM T36557 C4W5IY 16110419 EC50 = 4.2 nM T36557 CHJ4Z3 16110420 EC50 = 6.7 nM T36557 C2TO3Q 16110421 EC50 = 6.6 nM T36557 C2KPE7 16110422 EC50 = 43 nM T36557 CE16PQ 16110423 EC50 = 67 nM T36557 CDVL80 16110424 EC50 = 4.6 nM T36557 C3X2WM 16110425 EC50 = 25 nM T36557 C4T0RO 16110426 EC50 = 7.5 nM T36557 CT78IG 16110427 EC50 = 14 nM T36557 CYZ74P 16110428 EC50 = 11 nM T36557 C7IL6H 16110429 EC50 = 2230 nM T36557 CE91XP 16110436 EC50 = 5.9 nM T36557 C9W4KS 16110437 EC50 = 3.8 nM T36557 C2OZJ4 16110438 EC50 = 1.5 nM T36557 C6FA1K 16110439 EC50 = 2.3 nM T36557 CI05UK 16110440 EC50 = 43 nM T36557 CI4Z8S 16110441 EC50 = 11 nM T36557 C2UJ6Y 16110442 EC50 = 5.6 nM T36557 CBW78Z 16110443 EC50 = 2.2 nM T36557 CE19FD 16110444 EC50 = 0.95 nM T36557 C7F0IX 16110482 EC50 = 1.6 nM T36557 C3PXV5 16110483 EC50 = 0.58 nM T36557 C5WZ4Y 16110484 EC50 = 2.7 nM T36557 CCM5G9 16110485 EC50 = 4.4 nM T36557 C0N6VP 16110486 EC50 = 11 nM T36557 C5NX0T 16110487 EC50 = 2.9 nM T36557 C7Q2PD 16110488 EC50 = 1.3 nM T36557 CC24LB 16110489 EC50 = 2.2 nM T36557 CNU63E 16110490 EC50 = 249999995 nM T36557 CHD61I 16110491 EC50 = 2.1 nM T36557 CQ0T9X 16110492 EC50 = 12 nM T36557 CF15DS 16110493 EC50 = 1.2 nM T36557 CTC3I5 16110494 EC50 = 2.3 nM T36557 CNS35L 16110511 EC50 = 8.9 nM T36557 CXQD14 16110512 EC50 = 13 nM T36557 CKSV19 16110513 EC50 = 7.3 nM T36557 C4TO1G 16110514 EC50 = 56 nM T36557 CKN05Q 16110515 EC50 = 117 nM T36557 CZ5RS7 16110516 EC50 = 2.4 nM T36557 CU1S0A 16110517 EC50 = 2.7 nM T36557 CO5D1F 16110518 EC50 = 2.2 nM T36557 CB8Q6G 16110519 EC50 = 367 nM T36557 CW4V2X 16110524 EC50 = 1.3 nM T36557 CT35DL 16110525 EC50 = 6.9 nM T36557 C4F5EU 16110532 EC50 = 28 nM T36557 C09TRM 16110533 EC50 = 4.6 nM T36557 CZ3AN2 16110534 EC50 = 3 nM T36557 CXN40P 16110535 EC50 = 5.4 nM T36557 C0KL4A 16220189 Ki = 0.00483 nM T36557 CE71MI 16220190 EC50 = 0.72 nM T36557 CR3C1Q 16222636 EC50 > 10000 nM T36557 C49IER 16722365 EC50 = 1 nM T36557 CD7L4Z 16726113 EC50 = 0.03 nM T36557 C92NRU 16727109 EC50 > 25000 nM T36557 C6RT7K 16735280 Ki = 0.62 nM T36557 CVE58L 16735504 Ki = 0.0102 nM T36557 CN6CU3 16739344 EC50 = 1975 nM T36557 CD65RZ 16742591 EC50 > 1000 nM T36557 C8LPX0 16747684 EC50 = 4000 nM T36557 C83AOY 17894227 Ki = 2 nM T36557 CFS4T7 17894542 EC50 = 10 nM T36557 CLE7Y9 18442898 EC50 = 4680 nM T36557 CT1CI8 18442899 EC50 = 2630 nM T36557 CY0L2U 18442903 EC50 = 1050 nM T36557 CF9BK7 18701962 Ki = 3.7 nM T36557 CP8GD2 18702001 Ki = 5 nM T36557 C2GN1I 18766436 EC50 = 90 nM T36557 C2C8VM 20765803 EC50 = 4000 nM T36557 C3G8NO 20765805 EC50 = 1400 nM T36557 CW3G2Y 20777233 EC50 = 110 nM T36557 C59GOH 20826996 EC50 = 13600 nM T36557 CV7UB3 21054981 EC50 = 1400 nM T36557 COLV42 21054982 EC50 = 2300 nM T36557 CP3RI0 21054984 EC50 = 800 nM T36557 C5BM3O 21055003 EC50 = 1400 nM T36557 CMGS41 21866827 EC50 = 30000 nM T36557 CU0IJ4 21928218 EC50 = 4.5 nM T36557 C2O4BZ 21928229 EC50 = 11 nM T36557 CV0MX1 22229246 EC50 = 9 nM T36557 CU6YG1 22229249 EC50 = 148 nM T36557 C02WAZ 22229253 EC50 = 20 nM T36557 C28MRJ 22229258 EC50 = 229 nM T36557 C5JU1E 22229269 EC50 = 150 nM T36557 CL01NF 22229275 EC50 = 2 nM T36557 C4L5TH 22229292 EC50 = 534 nM T36557 C3F2OH 22229300 EC50 = 5 nM T36557 CFA14C 22229314 EC50 = 2 nM T36557 CSAX56 22229323 EC50 = 3 nM T36557 CM93FV 22279993 EC50 = 2210 nM T36557 CGVR07 22280001 EC50 = 251 nM T36557 CE3OI9 22280016 IC50 = 586 nM T36557 C1BG7A 22280047 IC50 = 356 nM T36557 C1G2OH 22280062 IC50 = 120 nM T36557 C14YDT 22280073 IC50 = 20 nM T36557 CDQ0Y6 22280103 EC50 = 295 nM T36557 C0VET7 22280114 IC50 = 313 nM T36557 C7IW1Y 22280124 IC50 = 76 nM T36557 COA0S5 22280155 EC50 = 252 nM T36557 CZS5Q3 22280173 EC50 = 933 nM T36557 CVH3O8 22280178 IC50 = 10.4 nM T36557 CE5BX0 22280187 EC50 = 585 nM T36557 CDZB48 22280210 EC50 = 267 nM T36557 CK1ZY7 22504766 EC50 = 1390 nM T36557 C8CP4E 22504797 EC50 = 6360 nM T36557 C2P7OG 22504815 EC50 = 561 nM T36557 C5YBQ0 22504835 IC50 = 97 nM T36557 C5X6IB 22504843 IC50 = 37 nM T36557 CDK75I 22504857 IC50 = 81 nM T36557 CO0UC5 22504899 EC50 = 1610 nM T36557 CHD4Z0 22504917 IC50 = 23 nM T36557 CS0HE9 22727983 EC50 = 1900 nM T36557 CE06NF 22728012 EC50 = 60 nM T36557 CT38PB 23111732 EC50 = 3260 nM T36557 CL6AD8 23628247 EC50 = 70 nM T36557 CS26KY 23648476 EC50 = 631 nM T36557 CO6EC1 23648933 EC50 = 300 nM T36557 C18CXM 23656548 EC50 = 130 nM T36557 C6CZ1W 23661590 EC50 = 1800 nM T36557 CS8L7W 23661728 EC50 = 130 nM T36557 CT43OQ 23661729 EC50 = 50 nM T36557 C9H4WT 23686961 EC50 > 10000 nM T36557 CTE1N2 24748569 EC50 > 10000 nM T36557 C56SGF 24754924 EC50 = 1 nM T36557 CNBV74 24759099 EC50 = 10 nM T36557 CJB0Y5 24776380 EC50 = 6 nM T36557 CHE16V 24776381 EC50 = 8.1 nM T36557 C5NIJ8 24776382 EC50 = 16 nM T36557 C7EJ4W 24776383 EC50 = 828 nM T36557 C39FEM 24776384 EC50 = 67 nM T36557 C6WK3P 24776385 EC50 = 130 nM T36557 COI0Q1 24776386 EC50 = 8 nM T36557 CPI7B6 24776387 EC50 = 24 nM T36557 CMA17V 24776388 EC50 = 40 nM T36557 CV4CJ0 24776389 EC50 = 286 nM T36557 CL1MV5 24776390 EC50 = 6.2 nM T36557 C5J2IY 24776391 EC50 = 29 nM T36557 CC1XW3 24776392 EC50 = 18 nM T36557 C3RCM7 24776393 EC50 = 67 nM T36557 C5N0IX 24776394 EC50 = 19 nM T36557 C73QEI 24808475 EC50 = 2.6 nM T36557 C15NSJ 24828803 EC50 > 30000 nM T36557 CO31MA 24828805 EC50 > 30000 nM T36557 CW51RK 24828806 EC50 > 100000 nM T36557 C3E7IZ 24882613 EC50 = 220 nM T36557 CP1EM0 24890166 EC50 = 210 nM T36557 C34OKV 24890167 EC50 = 4100 nM T36557 C0PYD9 24890168 EC50 > 10000 nM T36557 C5Q1GX 24890333 EC50 = 940 nM T36557 C5FV9O 24890334 EC50 = 550 nM T36557 C0P4RE 24890336 EC50 = 59 nM T36557 CMU63N 24890509 EC50 = 2200 nM T36557 CF57SZ 24890510 EC50 = 20 nM T36557 C13XCE 24890511 EC50 = 1400 nM T36557 C94RLU 24890513 EC50 = 45 nM T36557 C7LTC8 24890684 EC50 = 810 nM T36557 C3MDU5 24890685 EC50 = 6.8 nM T36557 C8PD2Z 24941254 IC50 = 125.89 nM T36557 C1P6WN 24949595 EC50 = 800 nM T36557 C17UHS 24949596 EC50 = 300 nM T36557 C1CG8I 24949919 EC50 = 700 nM T36557 CQWZ49 25032861 EC50 > 10000 nM T36557 CF98EG 25071332 EC50 = 25 nM T36557 CF3DZ4 25112371 EC50 = 43 nM T36557 CX97GA 25164959 IC50 > 50000 nM T36557 C45WHD 25165162 IC50 > 50000 nM T36557 CZF5B0 25165359 IC50 > 50000 nM T36557 C7W3IH 25165560 IC50 > 50000 nM T36557 CZ4TN9 25165638 IC50 > 50000 nM T36557 CER49X 25165639 IC50 > 50000 nM T36557 CBPX25 25166738 IC50 > 50000 nM T36557 C3HAY5 25166740 IC50 > 50000 nM T36557 C4WNU0 25166741 IC50 > 50000 nM T36557 CPE1I4 25166743 IC50 > 50000 nM T36557 CS03PW 25166956 IC50 > 50000 nM T36557 C64FTI 25211572 IC50 > 50000 nM T36557 CT51NS 25211876 EC50 = 12.59 nM T36557 CSWB02 25211877 EC50 = 15.85 nM T36557 C50YNC 25243830 EC50 = 120 nM T36557 CR3E5T 25263358 EC50 > 10000 nM T36557 CU68GV 25263359 EC50 = 199.53 nM T36557 COFY03 25263360 IC50 = 8 nM T36557 CL6SG8 25263361 EC50 = 199.53 nM T36557 CJW5Z8 25263362 IC50 = 25 nM T36557 C2YU5K 25263363 IC50 = 5 nM T36557 CB70OD 25263364 EC50 = 158.49 nM T36557 CE7MW2 25263365 EC50 > 10000 nM T36557 CAM4D7 25263366 IC50 = 13 nM T36557 C5KJS4 25263367 IC50 = 19.95 nM T36557 CT5R1F 25263368 IC50 = 3.999 nM T36557 CO16NL 25263369 IC50 = 10 nM T36557 C6NSB5 25263370 IC50 = 10 nM T36557 C7KPY3 25263371 IC50 = 15.85 nM T36557 CLS1I8 25263372 EC50 = 794.33 nM T36557 C7U4IG 25263373 IC50 = 15.85 nM T36557 CJ7NW1 25263374 EC50 = 19.95 nM T36557 CY09AD 25263375 IC50 = 10 nM T36557 CPT2M7 25263376 IC50 = 10 nM T36557 C3J6IA 25263377 IC50 = 10 nM T36557 CJG62V 25263378 IC50 = 20 nM T36557 CV5S1G 25263379 IC50 = 158 nM T36557 C5QA6B 25263380 IC50 = 10 nM T36557 CF49OS 25263381 IC50 = 62.95 nM T36557 CZDA26 25263382 IC50 = 31.99 nM T36557 CG59MP 25263383 IC50 = 3.981 nM T36557 CD9EZ2 25263384 IC50 = 16 nM T36557 C10NLX 25263385 EC50 = 630.96 nM T36557 C50GAO 25263386 IC50 = 5.998 nM T36557 C8KCW3 25263387 IC50 = 13 nM T36557 CJST96 25263388 EC50 = 100 nM T36557 CW6U1B 25263389 EC50 > 500 nM T36557 CKMR46 25263390 EC50 = 249 nM T36557 CZ0CO2 25263391 EC50 > 10000 nM T36557 C3P9KJ 25263392 EC50 = 720 nM T36557 CA8JG2 25263393 EC50 > 10000 nM T36557 C9B0PG 25263394 EC50 = 200 nM T36557 CE35MH 25263395 EC50 = 970 nM T36557 C3RG0W 25263396 EC50 = 560 nM T36557 C19DVJ 25263397 EC50 = 1070 nM T36557 C3FGA6 25263398 EC50 = 90 nM T36557 C04WDJ 25263399 EC50 = 50 nM T36557 CHL2X3 25263400 EC50 = 60 nM T36557 CNU8Q0 42608446 Ki = 5 nM T36557 CX70AK 42625720 EC50 > 10000 nM T36557 CW36AR 42625721 EC50 > 10000 nM T36557 CX6D9E 42625795 EC50 > 10000 nM T36557 C2TK3Z 42625796 EC50 > 10000 nM T36557 CRLG64 42625797 EC50 > 10000 nM T36557 C3UKN7 42625798 EC50 = 5270 nM T36557 CNE6U4 42625799 EC50 > 10000 nM T36557 CVAN68 42625871 EC50 > 10000 nM T36557 CG8K1S 42625874 EC50 > 10000 nM T36557 C86XNA 42625875 EC50 > 10000 nM T36557 CW0A6E 42625952 EC50 > 10000 nM T36557 C67UGQ 42625953 EC50 > 10000 nM T36557 CC6YK7 42625954 EC50 > 10000 nM T36557 C83VLK 42625955 EC50 > 10000 nM T36557 CC81PK 42625956 EC50 > 10000 nM T36557 C04ROU 42626028 EC50 = 4450 nM T36557 CI4VG0 42626029 EC50 > 10000 nM T36557 CIJ3H9 42626030 EC50 > 10000 nM T36557 CUS7L8 44132498 EC50 > 10000 nM T36557 CQ83EC 44143316 Ki = 8 nM T36557 C12XUE 44143317 Ki = 4 nM T36557 CD2VC6 44143318 Ki = 11 nM T36557 CBOX40 44143319 Ki = 16 nM T36557 C1GQC6 44143320 Ki = 35 nM T36557 C9FRI3 44143321 Ki = 36 nM T36557 C3DGV4 44143322 Ki = 47 nM T36557 C0Z8NG 44143323 Ki = 70 nM T36557 C6GJU8 44143324 Ki = 270 nM T36557 CK25QY 44143325 EC50 > 10000 nM T36557 C9D6TL 44143326 Ki = 7 nM T36557 C7U1JB 44143327 Ki = 6 nM T36557 C4OBI5 44143328 Ki = 22 nM T36557 C3ZL5T 44143329 Ki = 2 nM T36557 CX8Z3J 44143330 Ki = 0.6 nM T36557 CO72BR 44143331 Ki = 6 nM T36557 CZ3GO9 44143332 Ki = 9 nM T36557 C78CKO 44143333 Ki = 4 nM T36557 CLUG09 44143334 Ki = 16 nM T36557 C6VE7C 44143335 Ki = 35 nM T36557 CZF3A7 44143336 Ki = 120 nM T36557 C0UKO6 44143337 Ki = 36 nM T36557 CF2O9K 44143338 Ki = 28 nM T36557 CUG16K 44143339 Ki = 11 nM T36557 C4MB2X 44143340 Ki = 660 nM T36557 C7BS4Z 44143341 Ki = 1200 nM T36557 CNA0F7 44143342 Ki = 150 nM T36557 CM3N5P 44143343 Ki = 120 nM T36557 C5A4HL 44273874 EC50 = 2000 nM T36557 CE58NO 44273875 EC50 > 10000 nM T36557 CMX75T 44273944 EC50 = 1100 nM T36557 C0XNR5 44273963 EC50 = 4000 nM T36557 CC06QB 44273964 EC50 > 10000 nM T36557 CXOQ47 44274021 EC50 > 10000 nM T36557 CBY28T 44274044 EC50 > 10000 nM T36557 CNV3P0 44274047 EC50 > 10000 nM T36557 CH7M5T 44274107 EC50 > 10000 nM T36557 CM3SR4 44284994 EC50 = 5900 nM T36557 C67AKM 44316114 EC50 = 2500 nM T36557 C1HKA2 44316347 EC50 = 10000 nM T36557 CP3GE6 44316348 EC50 = 7900 nM T36557 C27PUY 44316349 EC50 = 1600 nM T36557 C1V6UE 44316496 EC50 = 2500 nM T36557 CX1V8Q 44316506 EC50 = 1600 nM T36557 CX07YR 44316521 EC50 = 500 nM T36557 C1LBQ7 44316568 EC50 = 160 nM T36557 CI19KT 44316591 EC50 = 7900 nM T36557 CNG0H5 44316592 EC50 = 500 nM T36557 C64ETY 44316824 EC50 = 790 nM T36557 CLQ0B3 44316825 EC50 = 4000 nM T36557 CKC5F4 44316880 EC50 = 500 nM T36557 CFT53Z 44316903 EC50 = 100 nM T36557 C3E7QU 44320897 EC50 = 900 nM T36557 CIY30P 44320978 EC50 = 2200 nM T36557 C6J0GY 44321201 EC50 = 3400 nM T36557 CLBK38 44321284 EC50 = 600 nM T36557 C4IR1A 44321440 EC50 = 5700 nM T36557 C45WMS 44321441 EC50 = 3400 nM T36557 CR3T1Q 44321462 EC50 = 2000 nM T36557 C9AEI4 44321463 EC50 = 700 nM T36557 CRFU18 44321490 EC50 = 1000 nM T36557 CH6Z2D 44321548 EC50 = 2200 nM T36557 C6ZK4E 44321572 EC50 = 400 nM T36557 CQ3RA9 44321573 EC50 = 2000 nM T36557 C6HM2Z 44321655 EC50 = 8300 nM T36557 C8N7LP 44331667 EC50 = 1000 nM T36557 CRG71X 44331668 EC50 = 93 nM T36557 CR9E3N 44331685 EC50 = 160 nM T36557 CTFW53 44331750 EC50 = 1000 nM T36557 CRNL38 44331751 EC50 = 430 nM T36557 CA36CR 44339522 IC50 > 15000 nM T36557 CV3R2S 44339547 IC50 > 15000 nM T36557 CZ25OL 44344272 EC50 = 3090 nM T36557 C9C8FN 44344313 EC50 = 3160 nM T36557 CWD8B7 44344585 EC50 = 3620 nM T36557 CU6HZ2 44345963 EC50 = 2400 nM T36557 CS3C7W 44365532 IC50 = 1500 nM T36557 CZ5BG6 44383664 Ki = 165 nM T36557 CK9PD5 44383828 Ki = 317 nM T36557 CIVC76 44383831 Ki = 529 nM T36557 CMB3S2 44383889 Ki = 37.5 nM T36557 C5ND3Y 44384224 Ki > 14000 nM T36557 CW9LD2 44384226 Ki = 203 nM T36557 CPY0K6 44384403 Ki = 156 nM T36557 CD4KM5 44384407 Ki = 18 nM T36557 C53DOZ 44384408 Ki = 3520 nM T36557 CTJD81 44384415 Ki = 26 nM T36557 CKDS82 44384419 Ki = 23 nM T36557 CA7YK9 44384460 Ki = 265 nM T36557 C4W7VN 44384466 Ki = 47 nM T36557 C46RVE 44384539 Ki = 47 nM T36557 C6PIU9 44384589 Ki = 136 nM T36557 C4R6EW 44384639 Ki = 4.6 nM T36557 CM8AE6 44385177 Ki = 62 nM T36557 C2FQX7 44385248 Ki = 508 nM T36557 CFM56P 44385352 Ki = 52 nM T36557 CE47ZL 44385396 Ki = 110 nM T36557 C6H0OL 44385399 Ki = 21 nM T36557 CY2O5S 44385405 Ki = 11 nM T36557 CH9UP4 44385406 Ki = 38 nM T36557 CRWI98 44386508 EC50 = 3 nM T36557 CDN54E 44388167 IC50 > 15000 nM T36557 C50FPR 44388210 IC50 = 4100 nM T36557 C5DNU7 44388563 IC50 > 50000 nM T36557 C51XZF 44388650 IC50 > 50000 nM T36557 C8E1NU 44388684 IC50 > 50000 nM T36557 CA1XK7 44388810 IC50 > 15000 nM T36557 CU1Y8L 44388819 IC50 > 15000 nM T36557 CU71OL 44388848 IC50 > 50000 nM T36557 C28TPK 44388866 IC50 > 15000 nM T36557 CMQ25R 44388882 IC50 = 7400 nM T36557 CQ6Z4Y 44388907 IC50 > 15000 nM T36557 CBV25F 44388914 IC50 = 13995.87 nM T36557 C0EH5G 44388966 IC50 > 15000 nM T36557 CF7L8V 44388968 IC50 > 50000 nM T36557 C5V0PS 44389085 IC50 > 15000 nM T36557 C0S6QK 44389098 IC50 > 50000 nM T36557 C6GF3L 44389191 IC50 = 5000 nM T36557 C1UGI7 44389733 EC50 = 11000 nM T36557 COXA71 44389801 EC50 = 18000 nM T36557 CX5A2Z 44389847 EC50 = 1900 nM T36557 C78VSM 44392315 IC50 = 1506.61 nM T36557 CJ49RK 44403670 EC50 = 1 nM T36557 C7IJ5H 44405121 EC50 = 420 nM T36557 C9DPH1 44405989 EC50 > 100000 nM T36557 CH7SB9 44406073 EC50 > 100000 nM T36557 CDX97W 44407180 EC50 = 700 nM T36557 CU24FD 44407220 EC50 = 1000 nM T36557 CJO4I9 44407221 EC50 = 500 nM T36557 C7X4UM 44407224 EC50 = 2000 nM T36557 C3I7OD 44409044 IC50 = 2387.81 nM T36557 C82CKD 44409063 IC50 = 3270 nM T36557 CTA6G7 44409088 EC50 = 55 nM T36557 CWGR81 44409098 IC50 = 742 nM T36557 C29VWO 44409126 IC50 = 1090 nM T36557 C6TRF5 44409127 IC50 = 2414 nM T36557 CJ8A6M 44409131 IC50 = 4630 nM T36557 C6Y1XC 44409170 IC50 > 50 nM T36557 CEBA60 44409171 IC50 = 4070 nM T36557 CB02UG 44409181 EC50 = 284 nM T36557 CK45XW 44409199 EC50 = 2230 nM T36557 C90PQA 44409212 IC50 = 134 nM T36557 C51XIC 44409274 IC50 = 603 nM T36557 CAN69Y 44409279 IC50 > 70000 nM T36557 CH5B7Q 44409318 IC50 = 1170 nM T36557 CZI2T9 44409319 IC50 = 1130 nM T36557 C17ZLP 44409323 IC50 = 1340 nM T36557 C9D7YM 44409430 IC50 = 1350 nM T36557 CU30EB 44411547 EC50 = 60 nM T36557 CYER28 44411548 EC50 = 90 nM T36557 CBYE57 44411557 EC50 = 110 nM T36557 CWR6V3 44411558 EC50 = 30 nM T36557 C5IWC6 44411561 EC50 = 40 nM T36557 C8G1HJ 44411562 EC50 = 560 nM T36557 CNO49B 44411563 EC50 = 210 nM T36557 C25NTU 44411565 EC50 = 60 nM T36557 C3G2CA 44411571 EC50 = 70 nM T36557 C4W6DO 44411577 EC50 = 40 nM T36557 CFB63G 44411578 EC50 > 10000 nM T36557 CM0RU6 44411581 EC50 = 70 nM T36557 COB80S 44411616 EC50 = 30 nM T36557 C4C9LD 44411618 EC50 > 10000 nM T36557 CY8K9S 44411630 EC50 > 10000 nM T36557 CNL81R 44411653 IC50 = 4 nM T36557 CW3AV8 44411661 IC50 = 7.998 nM T36557 C5P4BM 44411708 EC50 = 160 nM T36557 C5AR4E 44411737 EC50 = 350 nM T36557 C06BPM 44411740 EC50 = 490 nM T36557 C2G1LB 44411741 EC50 = 110 nM T36557 CQL2Z4 44411767 EC50 = 30 nM T36557 C2KCO7 44411772 EC50 = 540 nM T36557 C4MAN2 44411789 IC50 = 8600 nM T36557 C8FBH9 44411838 IC50 = 49 nM T36557 C4U2SJ 44411842 IC50 = 309.74 nM T36557 CJF9L1 44411843 IC50 = 88 nM T36557 CV3N5O 44411918 EC50 = 970 nM T36557 CFU5X3 44411943 EC50 = 110 nM T36557 CP1AZ6 44411945 EC50 = 50 nM T36557 C70NKQ 44411946 EC50 = 560 nM T36557 C71ZSM 44411968 EC50 = 70 nM T36557 CX6DN0 44411977 IC50 = 93 nM T36557 CP46GF 44412005 IC50 = 1400 nM T36557 CBVJ21 44412006 IC50 = 540 nM T36557 C8DPK5 44412188 IC50 = 39 nM T36557 CPK6G2 44412195 IC50 = 150 nM T36557 C1GH3B 44414891 EC50 = 3670 nM T36557 CU8NQ5 44414900 EC50 = 190 nM T36557 CKM0I8 44414901 EC50 = 30 nM T36557 C7LCH5 44414917 EC50 = 90 nM T36557 CBQ62J 44414926 EC50 = 2590 nM T36557 C07VTH 44414927 EC50 = 30 nM T36557 C1ETO8 44414955 EC50 > 10000 nM T36557 CV8IA5 44414956 EC50 > 10000 nM T36557 CTK8Z0 44414962 EC50 = 260 nM T36557 C1G4OC 44414967 EC50 = 310 nM T36557 C64UOB 44414968 EC50 = 110 nM T36557 CLO83A 44414991 EC50 = 130 nM T36557 C23ARN 44415004 EC50 = 4 nM T36557 C0TI2L 44415602 EC50 = 16 nM T36557 C4ZDC7 44415616 EC50 = 7 nM T36557 C04EOY 44415664 EC50 = 457 nM T36557 CVH8O0 44415665 EC50 = 1046 nM T36557 CPV1B6 44415695 EC50 = 10000 nM T36557 C1UO6R 44415696 EC50 = 82 nM T36557 C6C0YB 44415715 EC50 = 98 nM T36557 C9NB7J 44419009 EC50 > 10000 nM T36557 C97QXT 44419013 EC50 = 660 nM T36557 CBWX49 44420565 EC50 = 3021 nM T36557 CH1R7M 44420600 EC50 = 2.7 nM T36557 CL86VI 44424582 EC50 = 15 nM T36557 CV8X0N 44424583 EC50 = 4.8 nM T36557 C4QN7D 44424584 EC50 = 110 nM T36557 CK89CE 44424585 EC50 = 21 nM T36557 CNS39L 44424586 EC50 = 1.7 nM T36557 CGCJ17 44424587 EC50 = 1.9 nM T36557 C6LXQ5 44424588 EC50 = 8.3 nM T36557 CBZ1C3 44424589 EC50 = 3000 nM T36557 CBZU45 44424590 EC50 = 210 nM T36557 CC32AV 44424591 EC50 = 120 nM T36557 CQ1KL3 44424592 EC50 = 700 nM T36557 CG1CE6 44424593 EC50 = 40 nM T36557 CL2K0C 44424594 EC50 = 220 nM T36557 CSGM27 44424595 EC50 = 5.1 nM T36557 C30EJO 44425850 EC50 = 79 nM T36557 CQ9RH6 44425851 EC50 = 18.8 nM T36557 CH13TY 44425852 EC50 = 4.3 nM T36557 CGE39L 44425853 EC50 = 7 nM T36557 CX39CR 44425854 EC50 = 3.9 nM T36557 CBJU72 44425855 EC50 = 6.3 nM T36557 C3QLV7 44425856 EC50 = 70 nM T36557 CZ3X6Y 44425859 EC50 = 126 nM T36557 CN8A9Y 44425862 EC50 = 62.1 nM T36557 CP7JN9 44425864 EC50 = 7.4 nM T36557 CP6SO9 44425869 EC50 = 24.3 nM T36557 CDVH71 44425872 EC50 > 3000 nM T36557 CV6H9Z 44432125 IC50 = 62 nM T36557 CP0VK2 44432126 IC50 = 111 nM T36557 CORG53 44432127 IC50 = 286 nM T36557 C7L1WG 44432395 IC50 = 14 nM T36557 C06KRB 44432398 IC50 = 237 nM T36557 CWDS06 44432399 IC50 = 58 nM T36557 C9YZ1I 44432400 IC50 = 244 nM T36557 CK6PU9 44432401 IC50 = 42.95 nM T36557 CSF09X 44432402 EC50 = 166 nM T36557 CE51LN 44432403 IC50 = 3.597 nM T36557 CDV5O8 44432404 EC50 = 3120 nM T36557 CN7KJ9 44432405 IC50 = 24.1 nM T36557 CMO9I5 44432406 IC50 = 81 nM T36557 CA7OU6 44432407 IC50 = 6.8 nM T36557 C12ANM 44432408 IC50 = 734 nM T36557 CQ1W3L 44432409 EC50 = 254 nM T36557 C8AQ3I 44432410 IC50 = 91 nM T36557 CJ7GY1 44432411 EC50 = 4 nM T36557 CI45BS 44432832 EC50 = 160 nM T36557 CRPF69 44432835 EC50 = 11 nM T36557 CKHL98 44432837 EC50 > 10000 nM T36557 CD9C1K 44432838 EC50 = 770 nM T36557 CXR1O2 44432841 EC50 = 240 nM T36557 CEN1Z6 44432844 EC50 = 130 nM T36557 C1RN4F 44432845 EC50 = 320 nM T36557 CA1GL7 44432846 EC50 = 2000 nM T36557 CLZF68 44432847 EC50 = 220 nM T36557 C0BO8H 44432848 EC50 = 490 nM T36557 C5C4HV 44432849 EC50 = 3000 nM T36557 C03XMA 44432850 EC50 > 10000 nM T36557 CPQ0G2 44432851 EC50 = 1200 nM T36557 C2D5YP 44432852 EC50 = 3900 nM T36557 CBC74Q 44432853 EC50 = 150 nM T36557 C1A9NX 44432854 EC50 = 290 nM T36557 CF3L8X 44432855 EC50 = 290 nM T36557 CKTE10 44432857 EC50 = 12100 nM T36557 CWF49O 44434337 EC50 = 95 nM T36557 C53YEQ 44434338 EC50 = 81 nM T36557 C74NKE 44434339 EC50 = 59 nM T36557 C43PNF 44434340 EC50 = 22 nM T36557 CGD7Q8 44434341 IC50 = 3 nM T36557 CQP74N 44434342 IC50 = 39.99 nM T36557 CVWA23 44434343 IC50 = 32 nM T36557 C0VAZ9 44434344 EC50 = 30 nM T36557 C5WY9B 44434345 IC50 = 4 nM T36557 CM4K1D 44434346 IC50 = 5.998 nM T36557 CKI70B 44434347 EC50 = 50 nM T36557 CH5JP2 44434348 EC50 = 376 nM T36557 CQW7J6 44434349 EC50 = 1878 nM T36557 CS31PG 44434350 EC50 = 96 nM T36557 CERT39 44434351 IC50 = 5.998 nM T36557 C4B8VJ 44434352 EC50 = 48 nM T36557 CM8VY6 44434353 EC50 = 119 nM T36557 C9IG2C 44434354 EC50 = 1300 nM T36557 C4SMI1 44434355 IC50 = 3 nM T36557 C3O2BF 44434356 IC50 = 3 nM T36557 CRBM37 44434357 IC50 = 4 nM T36557 CL2H8U 44434358 IC50 = 9 nM T36557 CB5U3S 44434359 IC50 = 5 nM T36557 C4K0FY 44434360 EC50 = 87 nM T36557 CIA86O 44434361 IC50 = 3 nM T36557 C2VG9W 44434362 IC50 = 5 nM T36557 CL5AH3 44439623 IC50 = 7.998 nM T36557 CF01IC 44439624 IC50 = 9 nM T36557 C64AHD 44439625 IC50 = 14 nM T36557 CIW8B5 44439626 EC50 = 15 nM T36557 C7YHU2 44439631 EC50 = 25 nM T36557 CL1XI5 44439632 IC50 = 13 nM T36557 CM6Q0Y 44439633 EC50 = 6 nM T36557 CBQ3V5 44439710 EC50 = 24 nM T36557 CUF6W1 44439711 EC50 = 9 nM T36557 CB1RK5 44439712 EC50 = 12 nM T36557 CQW59J 44439713 EC50 = 83 nM T36557 CUJP69 44439715 EC50 = 7 nM T36557 CK14PR 44439716 EC50 = 7 nM T36557 CL9U1M 44439718 EC50 = 41 nM T36557 C5O8ZX 44439719 EC50 = 7 nM T36557 CBM0E7 44439721 EC50 = 23 nM T36557 CR2VY5 44439724 EC50 = 25 nM T36557 CO7CV3 44439725 EC50 = 16 nM T36557 C2RNS5 44439726 EC50 = 2 nM T36557 CVS0Q5 44439729 EC50 = 11 nM T36557 CU0JA6 44439730 EC50 = 3 nM T36557 C1JAZ3 44440776 EC50 = 1100 nM T36557 CYOD04 44440777 EC50 = 1900 nM T36557 CIR27Y 44440779 EC50 = 8000 nM T36557 CG43HK 44440780 EC50 = 160 nM T36557 CNI45S 44440781 EC50 = 5000 nM T36557 CQ25AW 44440782 EC50 = 1100 nM T36557 CWO5C2 44440783 EC50 = 1900 nM T36557 C3-OCT 44440785 EC50 = 140 nM T36557 C6TMR4 44440786 EC50 = 1700 nM T36557 C03TVK 44440787 EC50 = 1400 nM T36557 C4NDM7 44440789 EC50 = 120 nM T36557 COI23R 44440790 EC50 = 110 nM T36557 C8TOE9 44440791 EC50 = 830 nM T36557 C4BQ1C 44440792 EC50 = 6500 nM T36557 CDZ45N 44440795 EC50 = 1300 nM T36557 CA7G3R 44440797 EC50 = 3 nM T36557 C1PQ7V 44440800 EC50 = 1610 nM T36557 CX3P1C 44440804 EC50 = 1660 nM T36557 C62VTF 44440805 EC50 = 1190 nM T36557 CWDC32 44440806 EC50 = 1570 nM T36557 CVP5E8 44440925 EC50 = 2810 nM T36557 CRS8Z5 44440928 EC50 = 4880 nM T36557 C9F4ME 44440929 EC50 = 940 nM T36557 C7Y9VT 44440930 EC50 = 1740 nM T36557 CZ1TD8 44440931 EC50 = 1360 nM T36557 CS62GT 44440932 EC50 = 2610 nM T36557 CA69YP 44440933 EC50 = 2550 nM T36557 CFX28B 44440934 EC50 = 1170 nM T36557 C8DP1Z 44440935 EC50 = 2970 nM T36557 CL1EQ2 44440936 EC50 = 390 nM T36557 CUJ8X0 44441213 EC50 = 20000 nM T36557 CRWN48 44441214 EC50 = 13000 nM T36557 CV6RK5 44441215 EC50 = 7900 nM T36557 CQ23GJ 44441216 EC50 = 6000 nM T36557 CX5M7Q 44441220 EC50 = 3000 nM T36557 CEP16Z 44441344 EC50 = 15000 nM T36557 C31WIL 44446245 EC50 > 10000 nM T36557 CI64WZ 44446247 EC50 > 10000 nM T36557 C6XIU3 44446250 EC50 > 10000 nM T36557 CHY27Q 44446252 EC50 > 10000 nM T36557 CE1S5F 44446255 EC50 > 10000 nM T36557 C9OGX2 44446257 EC50 > 10000 nM T36557 CI49YJ 44446258 EC50 > 10000 nM T36557 CSH1U8 44446260 EC50 > 10000 nM T36557 C7YSZ5 44446262 EC50 = 400 nM T36557 C9GMW7 44446263 EC50 > 10000 nM T36557 CIR02A 44446264 EC50 > 10000 nM T36557 C85TKY 44451190 EC50 = 20 nM T36557 C7PA9S 44454244 EC50 = 870 nM T36557 C84FIQ 44454301 EC50 = 250 nM T36557 CIE06L 44454336 EC50 = 720 nM T36557 CP8OE3 44454364 EC50 = 360 nM T36557 CA84BK 44454366 EC50 = 8100 nM T36557 CLUF89 44458859 IC50 = 20 nM T36557 CC86GW 44458943 EC50 = 12 nM T36557 CR5SI0 44476535 EC50 > 10000 nM T36557 CU7GD5 44561770 IC50 > 50000 nM T36557 CPW0S4 44561816 IC50 > 50000 nM T36557 C9L3VY 44561817 IC50 > 50000 nM T36557 C08NKI 44561969 IC50 > 50000 nM T36557 CS48WU 44562841 EC50 > 25000 nM T36557 C94SYK 44562842 EC50 > 25000 nM T36557 C2RJ7Q 44568838 Ki = 2.54 nM T36557 CO5RI6 44587736 EC50 = 280 nM T36557 C15RIM 44587737 EC50 = 94 nM T36557 CVI68J 44587738 EC50 = 60 nM T36557 CO3IQ1 44587769 EC50 = 55 nM T36557 CNI3D6 44587770 EC50 = 28 nM T36557 CW67EM 44587801 EC50 = 180 nM T36557 C68RUE 44591751 EC50 = 117 nM T36557 C08IUA 44591752 EC50 = 45 nM T36557 CY59XQ 44591802 EC50 = 2710 nM T36557 C0S2NU 44591803 EC50 = 169 nM T36557 CN3WH7 44591815 EC50 = 137 nM T36557 CL6FI5 44591830 EC50 > 10000 nM T36557 CH9CK4 44626477 EC50 = 10 nM T36557 CPW57V 44626478 EC50 = 650 nM T36557 CUY95T 44626479 EC50 = 10 nM T36557 CI31DJ 44626480 EC50 = 10 nM T36557 C8TD4Z 44626481 EC50 = 10 nM T36557 C0Z3XM 44626583 EC50 = 5670 nM T36557 C3VF6I 44626585 EC50 = 1410 nM T36557 C3ME5P 44626586 EC50 = 110 nM T36557 CDIP96 44626587 EC50 = 70 nM T36557 C6V4SD 44626689 EC50 = 100 nM T36557 CB0GJ9 44626691 EC50 = 470 nM T36557 CP9YH7 44626696 EC50 = 331 nM T36557 C01AMG 44626697 EC50 = 160 nM T36557 CY3I4V 44626789 EC50 = 120 nM T36557 CXI58P 44626791 EC50 = 660 nM T36557 C4JRP9 44626797 EC50 = 56 nM T36557 C3YK1M 44626798 EC50 = 120 nM T36557 C3Q2XF 44626799 EC50 = 32 nM T36557 CB1ZX0 44626800 EC50 = 35 nM T36557 C4A0WS 44626801 EC50 = 26 nM T36557 CC08FO 44626884 EC50 = 9 nM T36557 C6N8RL 44626885 EC50 = 11 nM T36557 C3GX1Q 44626886 EC50 = 9 nM T36557 CEOS62 44626887 EC50 = 14 nM T36557 C6EF1Q 44626888 EC50 = 18 nM T36557 C6X8KS 44626889 EC50 = 63 nM T36557 C5I8NM 44626890 EC50 = 10 nM T36557 C8V9SP 44626891 EC50 = 31 nM T36557 CTY31Z 44626892 EC50 = 17 nM T36557 C4KC0Q 44626981 EC50 = 6 nM T36557 C53WQC 44626982 EC50 = 9 nM T36557 CQI69K 44626986 EC50 = 13 nM T36557 C8NAD5 44626987 EC50 = 30 nM T36557 C0RAL3 44626988 EC50 = 410 nM T36557 C4BNA9 44626989 EC50 = 52 nM T36557 CQ5O3I 44626990 EC50 = 45 nM T36557 CESB05 44627078 EC50 > 10000 nM T36557 CSW84C 44627079 EC50 > 10000 nM T36557 C3ZM7B 44627080 EC50 > 10000 nM T36557 C6B2RO 44627083 EC50 = 775 nM T36557 C2JB5Y 44627084 EC50 = 544 nM T36557 CABC27 44627085 EC50 = 23 nM T36557 CPS63M 44627086 EC50 = 2 nM T36557 CX41JP 44627087 EC50 = 6 nM T36557 CL34OS 44627188 EC50 = 3 nM T36557 CCQ59P 44627190 EC50 = 4 nM T36557 CMG9Q4 44627191 EC50 = 68 nM T36557 C9OI6W 44627192 EC50 = 59 nM T36557 CQJ26Z 44627297 EC50 > 10000 nM T36557 C87MHR 44627298 EC50 = 4060 nM T36557 C5W3IT 44627299 EC50 = 4710 nM T36557 CS25FR 44627300 EC50 = 6320 nM T36557 C0SYJ8 44627301 EC50 > 10000 nM T36557 CY49NK 44627302 EC50 = 34 nM T36557 C6RBQ1 44627303 EC50 = 8 nM T36557 CUL63M 44627304 EC50 = 6 nM T36557 C1G2QK 44627305 EC50 = 18 nM T36557 C96QCO 44627306 EC50 = 3 nM T36557 CR8A1I 44627407 EC50 = 320 nM T36557 CE2J5V 44627408 EC50 = 340 nM T36557 C43ZOX 44627409 EC50 = 1390 nM T36557 C7K0GI 44627410 EC50 = 2400 nM T36557 CA31WU 44627411 EC50 = 190 nM T36557 CPY46S 44627412 EC50 > 10000 nM T36557 CI1VN2 44627413 EC50 = 7 nM T36557 CK83HR 44627414 EC50 = 55 nM T36557 C1DQ7N 44627415 EC50 = 8 nM T36557 CF1Q5E 44627416 EC50 = 14 nM T36557 CPFN63 44627417 EC50 = 2 nM T36557 C9TNL0 44627524 EC50 = 130 nM T36557 C3OXU2 44627525 EC50 = 350 nM T36557 C3PZ6T 44627526 EC50 = 510 nM T36557 CD47HB 44627527 EC50 = 190 nM T36557 C1KAJ2 44627528 EC50 = 2620 nM T36557 CR93CX 44627529 EC50 = 1 nM T36557 CY95DP 44627531 EC50 = 930 nM T36557 CD8L4U 44627532 EC50 > 10000 nM T36557 CYJ52X 44627533 EC50 > 10000 nM T36557 CJ43OZ 44627627 EC50 = 5900 nM T36557 CEA3I2 44627628 EC50 = 130 nM T36557 CW7PG6 44627633 EC50 = 1200 nM T36557 CX0Q2Y 44627634 EC50 = 1870 nM T36557 CIWZ13 44627635 EC50 = 20 nM T36557 CA4W0L 44627636 EC50 = 2260 nM T36557 C28SEU 44627637 EC50 = 230 nM T36557 C6D0XF 44627728 EC50 = 60 nM T36557 CAQ41R 44627729 EC50 = 40 nM T36557 CCN8S2 44627730 EC50 = 70 nM T36557 CGO41A 44627731 EC50 = 140 nM T36557 C1HMU7 44627732 EC50 = 380 nM T36557 C8K3GF 44627733 EC50 = 2930 nM T36557 C3T1HB 44627734 EC50 = 740 nM T36557 CE93BG 44627735 EC50 = 340 nM T36557 CPFV72 44627838 EC50 > 10000 nM T36557 CEH41N 44627839 EC50 = 20 nM T36557 C2SJ5A 44627840 EC50 = 150 nM T36557 C53AJB 44627841 EC50 = 880 nM T36557 CXHP05 44627842 EC50 = 130 nM T36557 CZL75R 44627843 EC50 > 10000 nM T36557 CRI4Q6 44627844 EC50 = 460 nM T36557 CK7Z9X 44627845 EC50 = 1300 nM T36557 C95MPI 44627846 EC50 = 140 nM T36557 C8SPR5 44627847 EC50 = 480 nM T36557 C2LI9T 44627941 EC50 = 510 nM T36557 CA8CB6 44627942 EC50 = 720 nM T36557 CSDF01 44627943 EC50 = 10 nM T36557 CM5D8L 44627944 EC50 > 10000 nM T36557 CX23ZO 44627945 EC50 = 20 nM T36557 C35WJV 44627946 EC50 = 62 nM T36557 CP9G7C 44627948 EC50 = 1 nM T36557 C6JXF9 44628046 EC50 = 80 nM T36557 CQX2E8 44628047 EC50 = 50 nM T36557 CW2I4H 44628048 EC50 = 110 nM T36557 CUHD90 44628049 EC50 = 250 nM T36557 C24MHW 44628050 EC50 = 50 nM T36557 CI7SM1 45104339 IC50 = 100 nM T36557 C0OX9J 45104340 IC50 = 199.53 nM T36557 CB7ED5 45104341 IC50 = 1000 nM T36557 CLFU74 45104342 IC50 = 199.53 nM T36557 COD76Z 45104343 IC50 = 158.49 nM T36557 CGB9R5 45104439 IC50 = 125.89 nM T36557 CNEV35 45104440 IC50 = 125.89 nM T36557 CP7L6H 45104441 IC50 = 79.43 nM T36557 CF1Y2V 45104442 IC50 > 10000 nM T36557 C8L5CG 45104443 IC50 = 1258.93 nM T36557 CRIS28 45104444 IC50 > 10000 nM T36557 CTWC94 45104445 IC50 > 10000 nM T36557 C74OGR 45269453 EC50 = 11200 nM T36557 CQ4GE9 45273780 EC50 = 1400 nM T36557 CR46NQ 45375886 EC50 = 170 nM T36557 C72CNH 45783216 Ki = 5200 nM T36557 C89QTJ 46184983 EC50 > 50000 nM T36557 C5TUH7 46226812 Ki = 3.15 nM T36557 C25QHA 46226822 Ki = 2.98 nM T36557 CSR2C5 46226840 Ki = 2.37 nM T36557 C01JNB 46226841 Ki = 2.61 nM T36557 C2R8WH 46232959 EC50 > 10000 nM T36557 C12JOZ 46232960 EC50 > 10000 nM T36557 CL36PQ 46233001 EC50 > 10000 nM T36557 C3Q6DN 46233002 EC50 > 10000 nM T36557 C0P5ED 46233003 EC50 > 10000 nM T36557 C19XSC 46233038 EC50 > 10000 nM T36557 CBSA69 46233039 EC50 > 10000 nM T36557 C5O7FJ 46233040 IC50 > 10000 nM T36557 CE93XQ 46233070 IC50 > 10000 nM T36557 C9A2QS 46233071 EC50 > 10000 nM T36557 CT53DY 46233072 IC50 = 6950 nM T36557 CE72MC 46878644 EC50 = 70 nM T36557 C4WDX1 46878645 EC50 = 3200 nM T36557 C1QT8Z 46878727 EC50 > 10000 nM T36557 CWZ8N4 46878728 EC50 > 10000 nM T36557 C4WO1G 46878729 EC50 > 10000 nM T36557 CRK26D 46878777 EC50 = 3300 nM T36557 C0HYG2 46878778 EC50 = 6360 nM T36557 C49SRK 46878779 EC50 = 810 nM T36557 C62JTF 46878780 EC50 = 30 nM T36557 C3OZP9 46878781 EC50 = 18 nM T36557 C51RAC 46878843 EC50 = 250 nM T36557 CQ7JI0 46879867 EC50 = 29 nM T36557 CQF47Y 46879905 EC50 = 400 nM T36557 CAZ6N1 46879906 EC50 = 53 nM T36557 CDL01S 46880009 EC50 = 11 nM T36557 C8I4CV 46880010 EC50 = 45 nM T36557 C9T0FX 46880011 EC50 = 1.6 nM T36557 CFMH58 46880012 EC50 = 14 nM T36557 CQF9J7 46880049 EC50 = 4.9 nM T36557 CN9L7G 46916268 EC50 > 15000 nM T36557 CS13YQ 49846481 IC50 > 100000 nM T36557 CUD91T 49862248 EC50 > 10000 nM T36557 CP3Y0J 50925503 EC50 = 1 nM T36557 CD2G5X 50925504 EC50 = 1.8 nM T36557 C4PK6S 50942697 EC50 = 5 nM T36557 C96HOP 50942698 EC50 = 0.5 nM T36557 CK03LY 51038993 EC50 = 7200 nM T36557 CT59YM 51039006 EC50 = 2200 nM T36557 CX6BG9 51039007 EC50 = 750 nM T36557 CNVB53 51346913 EC50 = 800 nM T36557 CAXJ10 52918120 EC50 = 2.512 nM T36557 CRN19G 52918121 EC50 = 2.512 nM T36557 C3VEH4 52941520 EC50 = 220 nM T36557 C4KQR2 52948223 EC50 = 76 nM T36557 C2GE3H 52950020 EC50 = 5.7 nM T36557 CL83BY 53317593 EC50 = 7 nM T36557 CVN51I 53317892 EC50 = 4.5 nM T36557 CTUA27 53317893 EC50 = 6.2 nM T36557 C7I9UO 53319246 EC50 = 8.5 nM T36557 C1JIB3 53319416 EC50 = 25 nM T36557 CNWE60 53319417 EC50 = 2500 nM T36557 CPBS67 53322010 EC50 > 60000 nM T36557 C8JL7M 53323370 EC50 = 10 nM T36557 C1M8ZE 53323371 EC50 = 2000 nM T36557 CS2CX8 53324308 EC50 > 20000 nM T36557 C7L4BQ 53324689 EC50 = 1000 nM T36557 CX7H8M 53324690 EC50 = 500 nM T36557 C3PYV7 53325836 EC50 = 11 nM T36557 CB1OV9 53325996 EC50 = 1600 nM T36557 C79NKI 53325997 EC50 = 320 nM T36557 CL2VM8 54579977 IC50 = 158.49 nM T36557 CV9U5K 54580014 EC50 = 501.19 nM T36557 C9IN5X 54580015 EC50 = 125.89 nM T36557 C64SWC 54580016 EC50 = 125.89 nM T36557 C76WZO 54580529 EC50 = 1400 nM T36557 C6M9HP 54580530 EC50 = 580 nM T36557 CKBG47 54580531 EC50 = 800 nM T36557 CSH41U 54580814 EC50 = 2000 nM T36557 C8MLC0 54580964 EC50 = 1.995 nM T36557 C8EUF2 54580965 IC50 = 158.49 nM T36557 CM6I8P 54580966 EC50 = 316.23 nM T36557 CR5DC6 54580967 EC50 = 12.59 nM T36557 CPT96V 54581011 EC50 = 501.19 nM T36557 CM95BU 54581270 IC50 = 190.11 nM T36557 C81THX 54581535 EC50 = 300 nM T36557 CBE79V 54581857 EC50 = 1300 nM T36557 CAT03Y 54582018 EC50 = 25.12 nM T36557 CMLX87 54582047 EC50 = 794.33 nM T36557 CRKL15 54582795 EC50 = 5400 nM T36557 CT4IJ9 54582796 EC50 = 21 nM T36557 CQ89ZY 54582993 EC50 = 79.43 nM T36557 CP92OU 54582994 EC50 = 1000 nM T36557 CGTN92 54582995 EC50 = 1995.26 nM T36557 CHQ79P 54583754 EC50 = 6700 nM T36557 C1D5YV 54583795 EC50 = 9800 nM T36557 CK48SJ 54583995 EC50 = 63.1 nM T36557 C9YDX0 54583996 EC50 = 794.33 nM T36557 CX1V3U 54583997 IC50 = 7.943 nM T36557 CGXM65 54583998 EC50 = 3162.28 nM T36557 CK6CI7 54584935 EC50 = 398.11 nM T36557 C1KOF7 54584936 IC50 = 5011.87 nM T36557 CPXG09 54584937 EC50 = 1995.26 nM T36557 CBO34V 54584938 EC50 = 1258.93 nM T36557 CQU27M 54585710 EC50 > 10000 nM T36557 C4DX7E 54585711 EC50 = 700 nM T36557 C3TU7R 54585867 EC50 = 15.85 nM T36557 COX28A 54585896 EC50 = 316.23 nM T36557 C6ZSM0 54585897 EC50 = 501.19 nM T36557 CXL71T 54585898 EC50 = 316.23 nM T36557 C7D1LE 54585899 EC50 = 398.11 nM T36557 C0I2DH 54585900 EC50 = 501.19 nM T36557 CP8F9I 54585901 EC50 = 19.95 nM T36557 C0JOG1 54585902 EC50 = 39.81 nM T36557 C9Q0VG 54585903 EC50 = 31.62 nM T36557 CU43ME 54585904 EC50 = 39.81 nM T36557 CW0L9M 54586395 EC50 > 10000 nM T36557 C6EC0W 54586396 EC50 = 1400 nM T36557 CO0X2A 54586658 EC50 = 14900 nM T36557 CM9GL4 54586691 EC50 > 10000 nM T36557 C8NZ6D 54586832 EC50 = 158.49 nM T36557 C18JYB 54586833 IC50 = 63.1 nM T36557 C2K6FY 54586870 IC50 = 63.1 nM T36557 C8UO7K 54586871 EC50 > 10000 nM T36557 CTL0F5 54586872 EC50 = 6.31 nM T36557 C28UYH 54586873 EC50 = 39.81 nM T36557 C7N0YU 54587410 EC50 = 4800 nM T36557 C14QDZ 54587728 EC50 > 10000 nM T36557 C5J0BW 54587729 EC50 = 1200 nM T36557 C5ZX4B 54597874 EC50 > 10000 nM T36557 CRN5D3 54764927 EC50 = 55 nM T36557 CKIC64 56659331 EC50 = 11000 nM T36557 CRB95Z 56659332 EC50 = 3200 nM T36557 C92XSL 56659333 EC50 = 9700 nM T36557 CT1A3Y 56659334 EC50 = 1800 nM T36557 C4CP6U 56666265 EC50 = 14000 nM T36557 CIUN54 56666266 EC50 = 7300 nM T36557 C7NA3W 56666267 EC50 = 1900 nM T36557 CGP42W 56669681 EC50 = 4800 nM T36557 C5I0GB 56669682 EC50 = 2900 nM T36557 CH0KR3 56676514 EC50 = 62000 nM T36557 CQ58IX 56676515 EC50 = 25000 nM T36557 CN26ZO 56679837 EC50 = 13000 nM T36557 CXMR78 56925781 IC50 > 50000 nM T36557 C5HQZ6 56925892 IC50 > 50000 nM T36557 C0NRU5 56925893 IC50 > 50000 nM T36557 C2B6MF 56925894 IC50 > 50000 nM T36557 CJ46YQ 56925895 IC50 > 50000 nM T36557 CR6TP4 56925896 IC50 > 50000 nM T36557 CVO3A2 56925994 IC50 > 50000 nM T36557 CLCM62 56925995 IC50 > 50000 nM T36557 C8GLC1 56925996 IC50 > 50000 nM T36557 C2M8DR 56925997 IC50 > 50000 nM T36557 CD75ZU 56925998 IC50 > 50000 nM T36557 C8YGX7 56926094 IC50 > 50000 nM T36557 C15OKZ 56926095 IC50 > 50000 nM T36557 CN68DG 56926096 IC50 > 50000 nM T36557 C4K1XH 56926097 IC50 > 50000 nM T36557 CFO3R4 56926098 IC50 > 50000 nM T36557 C7X3WK 56926185 IC50 > 50000 nM T36557 CZEF98 56926186 IC50 > 50000 nM T36557 C92DPX 56926187 IC50 > 50000 nM T36557 CSJW15 56926188 IC50 > 50000 nM T36557 C9VTF3 56926189 IC50 > 50000 nM T36557 CMK92V 56926276 IC50 > 50000 nM T36557 CNB56J 56940812 EC50 = 1.6 nM T36557 CA7Y1Z 56941393 EC50 = 4.4 nM T36557 C1DQ4M 56942395 EC50 = 1.2 nM T36557 CN5Z9T 56945389 EC50 = 130 nM T36557 CNC6B5 56945390 EC50 = 570 nM T36557 CRJC63 56945487 EC50 = 850 nM T36557 C0MC8V 56949691 EC50 > 10000 nM T36557 CQ19IH 56949692 EC50 > 10000 nM T36557 CB4F9K 56949693 EC50 > 10000 nM T36557 CS0AP9 57342889 IC50 = 30.4 nM T36557 C9SB5K 57390812 EC50 = 7100 nM T36557 CIFN56 57391546 EC50 > 10000 nM T36557 C8Y0ET 57391547 EC50 > 10000 nM T36557 CT3U5R 57392587 EC50 > 8100 nM T36557 CIVL69 57392628 EC50 > 13000 nM T36557 CX8QN1 57392629 EC50 = 1900 nM T36557 C7A2XY 57392630 EC50 = 8800 nM T36557 C5JD9O 57392836 EC50 = 470 nM T36557 C5I1CA 57393296 EC50 > 10000 nM T36557 C5A7HW 57393297 EC50 > 10000 nM T36557 C5BG1A 57394147 EC50 = 290 nM T36557 CZ0Y1N 57394350 EC50 > 6800 nM T36557 CX34SN 57394351 EC50 > 11000 nM T36557 C7Q3IB 57395028 EC50 > 10000 nM T36557 CHRX78 57396101 EC50 = 3100 nM T36557 C9V1KC 57396779 EC50 > 10000 nM T36557 CQ71JU 57396780 EC50 > 10000 nM T36557 CLI70F 57396782 EC50 > 10000 nM T36557 C7YC4Z 57396783 EC50 > 10000 nM T36557 C2DOZ9 57397718 EC50 = 580 nM T36557 C3O8JG 57398546 EC50 > 10000 nM T36557 C6ET7R 57398547 EC50 > 10000 nM T36557 C1DPW9 57398548 EC50 > 10000 nM T36557 C19KAD 57398549 EC50 > 10000 nM T36557 CPV28C 57399559 EC50 > 17000 nM T36557 CQT4G5 57400212 EC50 > 10000 nM T36557 CQC7F9 57400214 EC50 > 10000 nM T36557 CXO3V1 57401284 EC50 > 13000 nM T36557 C82NSD 57401312 EC50 = 1800 nM T36557 CTWX97 57402017 EC50 > 10000 nM T36557 C69PVW 57403073 EC50 = 2400 nM T36557 CXA36C 57404419 EC50 = 47600 nM T36557 CS4J1B 57404439 EC50 = 48500 nM T36557 C1Y7WA 58754075 IC50 = 5.998 nM T36557 C79PXW 60166133 EC50 = 6.1 nM T36557 COCI72 60166134 EC50 = 38.8 nM T36557 CO2X7F 60166264 EC50 = 57.2 nM T36557 CY31AP 60166265 EC50 = 132 nM T36557 C38XJT 60166266 EC50 = 60 nM T36557 CFA9N8 60166267 EC50 = 9.4 nM T36557 CES4D2 60166268 EC50 = 4.8 nM T36557 C3P5MV 60166383 EC50 = 11.4 nM T36557 CR01ID 60166384 EC50 = 2.1 nM T36557 C6U3KL 60166385 EC50 = 1.2 nM T36557 CN78JU 60166386 EC50 = 2.8 nM T36557 C7IW2B 60166387 EC50 = 4.6 nM T36557 CC3HM4 60166513 EC50 = 6.7 nM T36557 CL0V6S 60166514 EC50 = 8.1 nM T36557 CON53Z 60166515 EC50 = 490.1 nM T36557 CZ8VU0 60166647 EC50 = 16.7 nM T36557 CYT71B 60166648 EC50 = 523 nM T36557 CG71ZE 60166649 EC50 = 1.8 nM T36557 CC4YD6 60166650 EC50 = 1 nM T36557 C3LGI6 60166651 EC50 = 1.1 nM T36557 CALX08 60166891 EC50 = 1.1 nM T36557 C9RO7Z 68588383 EC50 = 71.4 nM T36557 C1WL3P 68674744 EC50 = 1912 nM T36557 CS4V7A 68676158 EC50 > 5000 nM T36557 C9PF1U 68676459 EC50 = 1387 nM T36557 CH62WK 68676471 EC50 = 1230 nM T36557 CI7DX4 68676782 EC50 = 1098 nM T36557 CFN69J 68677403 EC50 = 645 nM T36557 CIYO07 68677705 EC50 > 5000 nM T36557 CIU96H 68677842 EC50 = 866 nM T36557 CY9GZ8 70681800 IC50 = 5 nM T36557 C2DZ3G 70681801 IC50 = 7227.7 nM T36557 CSEF42 70681805 IC50 = 891.25 nM T36557 CMT6J3 70681806 IC50 = 1510.08 nM T36557 CB4A7U 70683915 IC50 = 5069.91 nM T36557 C7TJC3 70686048 IC50 = 7040 nM T36557 C13CJK 70686054 IC50 = 3845.92 nM T36557 CEL43F 70688075 EC50 = 2.3 nM T36557 C40KCB 70688165 IC50 = 1499.68 nM T36557 CFY6Z4 70688166 IC50 = 160 nM T36557 CP72KL 70688172 IC50 = 372.39 nM T36557 CIC8V5 70690196 IC50 = 7.998 nM T36557 C69MGD 70692364 IC50 = 3499.45 nM T36557 C34KXB 70692371 IC50 = 920.45 nM T36557 CR2YQ9 70693621 EC50 = 51100 nM T36557 C5C9HR 70694419 IC50 = 3800 nM T36557 C4DRC8 70694428 IC50 = 139.96 nM T36557 C29DRB 70694429 IC50 = 169.82 nM T36557 CV3T4P 70695727 EC50 = 53100 nM T36557 CR2PJ4 70695728 EC50 = 33900 nM T36557 CL0JN8 70696489 IC50 = 6900 nM T36557 C90GXS 70696490 IC50 = 258.82 nM T36557 C9PA6Y 71449654 EC50 = 13100 nM T36557 CC5T1Z 71450448 EC50 = 6400 nM T36557 C2TLF8 71450909 EC50 = 2100 nM T36557 CM63BE 71452661 EC50 = 6900 nM T36557 C9ERN1 71453290 EC50 = 11000 nM T36557 CY7UG1 71454437 EC50 = 18000 nM T36557 C5US2A 71455005 EC50 = 30100 nM T36557 C8PBI3 71456242 EC50 = 2200 nM T36557 C9RB3Y 71459933 EC50 = 15000 nM T36557 C2LG7J 71459934 EC50 = 4100 nM T36557 CX1SC6 71461648 EC50 = 19000 nM T36557 CLN26W 71544843 EC50 = 23.7 nM T36557 CL4A2V 71604423 EC50 = 7 nM T36557 C10SPC 71616170 EC50 = 40 nM T36557 CNPK13 71616171 EC50 = 152 nM T36557 CI1LF2 71616173 EC50 = 16 nM T36557 C9U6VX 71616290 EC50 = 131 nM T36557 CK58CF 71616294 EC50 = 14 nM T36557 C6LT3W 71616409 EC50 = 328 nM T36557 C5NU0T 71721539 IC50 = 6000 nM T36557 CNR9P8 73347576 IC50 = 92 nM T36557 C9SET4 73350677 IC50 = 29 nM T36557 C8PVH7 73352177 IC50 = 28 nM T36557 C3ARC8 73352181 IC50 = 13 nM T36557 C23BML 73353639 IC50 = 19 nM T36557 C9PBS7 73356704 IC50 = 100 nM T36557 C32YPJ 76321033 EC50 = 79 nM T36557 CDY64J 76321238 IC50 > 30000 nM T36557 C6X5MD 86279340 EC50 = 4700 nM T36557 CK9IH1 86281822 EC50 = 9.8 nM T36557 CV82FO 87225689 EC50 = 78 nM T36557 C63WUO 87537807 EC50 = 919 nM T36557 C4BA8W 90656430 IC50 > 100000 nM T36557 CA9PL8 91663316 IC50 = 25 nM T36557 C7R6IK 101882290 EC50 = 3000 nM T36557 CA6I4Y 101896436 EC50 = 6400 nM T36557 CFCE51 101896437 EC50 = 1300 nM T36557 C1CN0A 117629817 EC50 = 13 nM T36557 C2NT4A 117940654 IC50 = 30 nM T36557 C8RZ0N 117940704 IC50 = 438 nM T36557 C2HMU9 117940709 IC50 = 515 nM T36557 C8M6VO 117940743 IC50 = 124 nM T36557 CAWZ74 117940820 IC50 = 18 nM T36557 C32XBP 117940859 IC50 = 47 nM T36557 C9BA5Q 117940874 IC50 = 40 nM T36557 CA95EY 117940949 IC50 = 66 nM T36557 CFYW64 117940962 IC50 = 1620 nM T36557 C0J6WT 117940970 IC50 = 667 nM T36557 C0R8BX 117940999 IC50 = 131 nM T36557 CG7F5W 117941020 IC50 = 138 nM T36557 C3UR2N 117941053 IC50 = 3590 nM T36557 C0VNL8 117941054 IC50 = 34 nM T36557 CWL20F 117941134 IC50 = 61 nM T36557 CHN6Z5 117941185 IC50 = 1240 nM T36557 C4F1NK 117941228 IC50 = 83 nM T36557 C9M7RL 118714598 EC50 = 3200 nM T36557 C49HBU 118714599 EC50 = 12000 nM T36557 CN4PU6 118714603 EC50 = 3000 nM T36557 CA1RT3 118714624 EC50 = 5400 nM T36557 C0PTU8 118720593 EC50 = 25000 nM T36557 CZP8E7 118725344 EC50 = 6300 nM T36557 CKC50A 118725345 EC50 = 3400 nM T36557 C5ENC7 118725346 EC50 = 2200 nM T36557 CTH73Y 118725347 EC50 = 6800 nM T36557 CQ4OY5 118725348 EC50 = 7400 nM T36557 C9M1BC 118725349 EC50 = 2300 nM T36557 CX5TV7 118725351 EC50 = 5900 nM T36557 CH5RB6 118734332 IC50 = 284 nM T36557 C4E3AX 121269371 EC50 = 5 nM T36557 CW23RD 121269378 EC50 = 690 nM T36557 C26PFK 121269380 EC50 = 1.93 nM T36557 C0Q8MC 121269381 EC50 = 1.59 nM T36557 C3AP2B 121269382 EC50 = 80 nM T36557 CX4AN2 121269406 EC50 = 1850 nM T36557 CMDE36 121269416 EC50 = 5.51 nM T36557 CLRU83 121269424 EC50 = 230 nM T36557 C0BZ5D 121269430 EC50 = 19.8 nM T36557 CL1O6E 121269470 EC50 = 13.49 nM T36557 C5FD2E 121277013 EC50 = 64.5 nM T36557 CC32JH 121277016 EC50 = 510 nM T36557 C0BKL7 121277018 EC50 = 82.5 nM T36557 CE3YL2 121277093 EC50 = 40 nM T36557 CPA8J7 121277097 EC50 = 210 nM T36557 C6TBD2 121345502 EC50 > 20000 nM T36557 C0BI8N 122183534 EC50 = 6300 nM T36557 CHYL24 122183546 EC50 = 9400 nM T36557 CM1S7B 122370046 EC50 = 320 nM T36557 C40QCP 125623112 EC50 > 100000 nM T36557 C9C0LW 127029850 EC50 = 175 nM T36557 C06KLU 127029851 EC50 = 920 nM T36557 C14GFR 127032530 EC50 > 10 nM T36557 C0P8LB 127033514 EC50 = 863 nM T36557 CCI7M6 127033818 EC50 = 218 nM T36557 CM64PE 127033821 EC50 = 264 nM T36557 C0MH3C 127034370 EC50 = 306 nM T36557 C0YG1M 127034508 EC50 = 1 nM T36557 CKQ3O5 127038041 IC50 = 320 nM T36557 CDF2I5 127039433 IC50 = 907 nM T36557 CP72EH 127039434 IC50 = 1431 nM T36557 CDV84X 131747741 EC50 > 20000 nM T36557 C1PGI4 132578432 EC50 = 390 nM T36557 C36ESP 132578434 EC50 = 290 nM T36557 C6W4KX 132578490 EC50 = 23 nM T36557 CX69BS 134139597 EC50 = 370 nM T36557 C0Y4CW 134154728 EC50 = 1000 nM T36557 CV6OP5 135513372 EC50 > 10000 nM T36557 CL6Q7I 136000613 EC50 = 900 nM T36557 C9IU2J 136088972 IC50 = 10 nM T36557 CW8QT1 137527725 IC50 > 75000 nM T36557 C7DS5O 137633219 EC50 = 1120 nM T36557 CYG4I2 137633420 EC50 = 2026 nM T36557 C15XNC 137637824 EC50 = 1650 nM T36557 C6LI3N 137637955 EC50 = 1259 nM T36557 C8FZ6W 137639177 EC50 = 31000 nM T36557 CI5ER2 137639724 EC50 = 1140 nM T36557 CSP9K7 137641115 EC50 = 1347 nM T36557 CBC61V 137647253 EC50 = 697 nM T36557 C93IRA 137648584 EC50 = 1607 nM T36557 CRB9Z7 137651528 EC50 > 5000 nM T36557 CJ6DS1 137654442 EC50 = 1600 nM T36557 CS43WD 137654739 EC50 = 1085 nM T36557 CLA1N3 137655653 EC50 = 320 nM T36557 CZ84GI 137655707 EC50 > 5000 nM T36557 CQI07K 137656641 EC50 = 990 nM T36557 CL1RG9 137659246 EC50 = 2100 nM T36557 COWM26 137659583 EC50 = 450 nM T36557 CUA42H 137660782 EC50 = 970 nM T36557 CC5X3V 139501076 EC50 = 38600 nM T36557 CFM9U6 139501078 EC50 > 100000 nM T36557 C5WRM9 139501186 EC50 > 100000 nM T36557 C9KYQ5 139501208 EC50 = 8900 nM T36557 CKS10N 145704693 EC50 = 810 nM T36557 CCF02H 145964530 IC50 = 6600 nM T36557 C56SHA 145964597 IC50 = 10900 nM T36557 C5DH4X 145964745 EC50 > 10000 nM T36557 C5H8EZ 145965425 IC50 = 11300 nM T36557 CPG7N1 145965467 EC50 > 10000 nM T36557 CC3X5W 145965684 EC50 = 11000 nM T36557 CFX4L5 145965707 EC50 > 10000 nM T36557 CB5Z9S 145965895 EC50 = 8700 nM T36557 C6BSE0 145965984 EC50 = 1400 nM T36557 CHP5B6 145970080 EC50 = 1090 nM T36557 CK1MR7 145972041 EC50 = 880 nM T36557 CX06DP 145974139 EC50 = 1800 nM T36557 C6QGN9 145975013 EC50 > 1000 nM T36557 CJDH32 145975435 EC50 = 270 nM T36557 CG1XZ6 145975539 EC50 = 2600 nM T36557 CUB0I8 145977098 EC50 = 4600 nM T36557 C4GQ3Y 145977517 EC50 > 1000 nM T36557 C98CHS 145977976 IC50 = 10900 nM T36557 C0KP3F 145980573 EC50 = 4840 nM T36557 C1Q6PV 145980608 EC50 = 1980 nM T36557 CKR43C 145981599 EC50 = 9570 nM T36557 C87UAM 145982210 EC50 = 1520 nM T36557 CFY8U2 145982433 EC50 = 1950 nM T36557 C4D7TZ 145982651 EC50 = 4.5 nM T36557 CT0YS3 145982746 EC50 = 9.5 nM T36557 C65PGI 145982771 EC50 = 7 nM T36557 CTFM01 145982798 EC50 = 12 nM T36557 C65FME 145983252 EC50 = 65 nM T36557 CH1XJ8 145983321 EC50 = 86 nM T36557 C3WJZ8 145983637 EC50 = 9.1 nM T36557 CP4W3R 145983705 EC50 = 4 nM T36557 CT90OW 145983779 EC50 = 25 nM T36557 CFJ94I 145984084 EC50 = 5.3 nM T36557 C8V7OD 145984577 EC50 = 10 nM T36557 C4LN8E 145984731 EC50 = 3.2 nM T36557 CIV2P1 145984795 EC50 = 56 nM T36557 C0C2SU 145984820 EC50 = 6.3 nM T36557 CTY5A8 145984841 EC50 = 0.7 nM T36557 CQ1TB7 145984906 EC50 = 2160 nM T36557 CCYK53 145985074 EC50 = 6.1 nM T36557 CV84PQ 145985229 EC50 = 5.8 nM T36557 CH9OI0 145985286 EC50 = 26 nM T36557 CG8R3L 145985481 EC50 = 6.9 nM T36557 C9LA1O 145985668 EC50 = 38 nM T36557 CRAK83 145985994 EC50 = 18 nM T36557 CAE95K 145986458 EC50 > 10000 nM T36557 CW7Y4G 145986696 EC50 = 1750 nM T36557 CBOR53 145986704 EC50 = 1930 nM T36557 C0G2WE 145988431 EC50 = 1730 nM T36557 C75DSN 145989198 EC50 = 2420 nM T36557 CI39OJ 145989913 EC50 = 7930 nM T36557 CJ76KD 145990303 EC50 = 5490 nM T36557 CV2FB6 145992078 EC50 = 2370 nM T36557 C6F0LJ 145992170 EC50 = 4560 nM T36557 CP79UQ 145992176 EC50 = 2090 nM T36557 CCV39B 145994196 EC50 = 3350 nM T36557 C7X3AL 153763221 EC50 = 17000 nM T36557 CD5QM6 155511861 EC50 = 5 nM T36557 C8Y9ST 155512244 EC50 = 1320 nM T36557 CJRW35 155512467 IC50 > 100000 nM T36557 C3Z6VL 155514089 EC50 = 13000 nM T36557 CDA4C9 155515667 IC50 = 820 nM T36557 CICX19 155516325 EC50 > 10000 nM T36557 C29DXN 155517010 EC50 = 2300 nM T36557 CS48YI 155517472 EC50 = 150 nM T36557 C08DTF 155517891 EC50 = 376 nM T36557 C2COG3 155517895 EC50 = 1800 nM T36557 C2C4OZ 155518329 EC50 > 10000 nM T36557 C1POU5 155518522 EC50 = 6200 nM T36557 C86OCS 155520630 IC50 = 610 nM T36557 C6R1TF 155520683 EC50 = 2800 nM T36557 C6EW5F 155523441 EC50 = 3900 nM T36557 C17OFD 155523655 EC50 = 2660 nM T36557 C3GH8U 155523815 EC50 > 100000 nM T36557 C4Q7TF 155524299 EC50 = 290 nM T36557 C4GEH1 155525496 IC50 = 3740 nM T36557 CPT9J8 155525700 EC50 = 780 nM T36557 CV51OZ 155526003 IC50 = 27730 nM T36557 C3P2ZK 155526024 EC50 > 10000 nM T36557 C95KYP 155526365 EC50 = 4300 nM T36557 CO7NR2 155528574 EC50 = 6500 nM T36557 C3LZQ1 155528955 EC50 = 1200 nM T36557 C34YXP 155529382 EC50 > 10000 nM T36557 C7NDX5 155529750 EC50 > 10000 nM T36557 C6N9YP 155530111 EC50 = 729 nM T36557 C9YTH8 155530420 EC50 > 10000 nM T36557 CT5D9K 155530726 EC50 > 10000 nM T36557 COG5A0 155530735 EC50 = 5700 nM T36557 C6W2JV 155531862 EC50 > 100000 nM T36557 C2O9VS 155532185 EC50 = 400 nM T36557 C63HSA 155534748 EC50 = 5 nM T36557 CE7I8Q 155534885 EC50 = 29000 nM T36557 C2FU1O 155535195 IC50 = 225 nM T36557 C0B5MT 155535253 EC50 = 400 nM T36557 CS86YB 155535303 EC50 = 3100 nM T36557 CVG6P0 155535946 EC50 > 10000 nM T36557 CR9BE4 155536793 IC50 = 1970 nM T36557 CHC04X 155536991 EC50 = 5300 nM T36557 CN48LF 155537424 EC50 = 110 nM T36557 CM7S9F 155537835 IC50 = 24970 nM T36557 CE2LR1 155538630 EC50 > 100000 nM T36557 C3R9YL 155539254 EC50 = 34000 nM T36557 C64FRG 155541703 IC50 = 319 nM T36557 CSI9G7 155541727 EC50 = 7000 nM T36557 CXI91F 155543520 IC50 = 22230 nM T36557 C5W8SV 155543683 EC50 > 10000 nM T36557 C1YSQ7 155545016 EC50 = 46 nM T36557 C6PD1A 155545127 EC50 = 972 nM T36557 CX3KF2 155545207 EC50 > 10000 nM T36557 CLH91J 155545920 IC50 = 439 nM T36557 C1PO2Q 155546331 EC50 > 10000 nM T36557 CNSF75 155546388 IC50 = 48800 nM T36557 CFQ28J 155546921 EC50 = 1100 nM T36557 CC63ZG 155547595 EC50 = 564 nM T36557 CR48CL 155547604 EC50 = 529 nM T36557 C2QGR5 155549327 EC50 = 6800 nM T36557 CZ59YK 155550531 IC50 = 197 nM T36557 C87TQJ 155551096 EC50 = 4300 nM T36557 C2MTF9 155552428 EC50 = 9200 nM T36557 CWG10F 155552953 IC50 = 4490 nM T36557 C3KD0I 155553701 IC50 = 79 nM T36557 C7IN4B 155554421 EC50 = 2800 nM T36557 CUAP95 155555299 EC50 > 10000 nM T36557 CJQ54R 155556924 EC50 = 11000 nM T36557 C4BSK6 155557354 EC50 = 1650 nM T36557 CVH06N 155560437 EC50 > 10000 nM T36557 CM52UW 155560868 EC50 = 7100 nM T36557 CQ6VH4 155561358 EC50 = 1160 nM T36557 CUDT29 155561763 IC50 = 25550 nM T36557 C2NPT3 155561834 EC50 > 10000 nM T36557 C37ZFX 155563228 EC50 = 436 nM T36557 CK94IU 155564010 IC50 = 2780 nM T36557 CG02XL 155565451 EC50 = 102 nM T36557 CEWX25 155565883 EC50 = 4100 nM T36557 C3FK2M 155566781 EC50 = 6100 nM T36557 CQP4Y0 155569313 EC50 = 1400 nM T36557 D00TFA 3392731 EC50 = 6200 nM T36557 D02TRN 445638 IC50 = 9600 nM T36557 D02TVS 985 IC50 = 7400 nM T36557 D02WFA 5281 IC50 = 6000 nM T36557 D03BPG 2777391 IC50 > 10000 nM T36557 D03LOG 5280450 IC50 = 10000 nM T36557 D05CLM 9870304 EC50 = 150 nM T36557 D06VBQ 46233311 IC50 = 155 nM T36557 D07MBC 5283454 EC50 = 1100 nM T36557 D08OBF 11005 IC50 = 24000 nM T36557 D08QXD 9935197 IC50 = 4 nM T36557 D08UWZ 16725047 EC50 > 25000 nM T36557 D08ZYC 11595431 Ki < 3162.28 nM T36557 D09JII 9891946 EC50 = 6 nM T36557 D09XCX 5694 EC50 = 1460 nM T36557 D0A4EA 445639 IC50 = 5300 nM T36557 D0C5SV 5280934 IC50 = 16000 nM T36557 D0E7NO 2969 IC50 = 30000 nM T36557 D0F0MP 9889841 EC50 = 11 nM T36557 D0HD9P 444899 IC50 = 3100 nM T36557 D0K1TQ 9934458 EC50 = 1 nM T36557 D0N0UC 3893 IC50 = 30000 nM T36557 D0NM0G 2800647 IC50 = 284 nM T36557 D0O2US 9870584 Ki = 1200 nM T36557 D0W7RI 5311242 EC50 = 1880 nM T36557 D0XR8Q 1517 EC50 = 190 nM T36557 D0YK9T 6603901 EC50 = 20 nM T69413 D01MXK 73167574 EC50 = 25100 nM T69413 CYG16X 215405 EC50 > 100000 nM T69413 CQV28T 806021 EC50 = 16400 nM T69413 C26FYK 883012 EC50 = 63000 nM T69413 CNBT48 886392 EC50 > 100000 nM T69413 CRTD92 940433 EC50 > 100000 nM T69413 C7SDM5 947638 EC50 > 100000 nM T69413 C23NCZ 1285085 EC50 = 9700 nM T69413 CO2U1S 1316842 EC50 > 100000 nM T69413 CPJ21O 1419434 EC50 > 100000 nM T69413 COI17W 3733580 EC50 = 23200 nM T69413 CTX17I 10734486 EC50 = 8600 nM T69413 CY64AR 11172250 EC50 > 100000 nM T69413 CI0T8W 39861393 EC50 > 100000 nM T69413 CD9VN0 39861419 EC50 > 100000 nM T69413 CLN30P 39861421 EC50 > 100000 nM T69413 CJFU79 39861427 EC50 > 100000 nM T69413 C0SQ4W 39861440 EC50 = 13100 nM T69413 C9S7AR 56700010 EC50 > 100000 nM T69413 CBF4Z2 70682681 IC50 = 25000 nM T69413 CTO5X9 73167576 EC50 >= 89700 nM T69413 CBY4N2 103041476 EC50 > 100000 nM T69413 C62BFY 117072009 EC50 > 100000 nM T69413 C2K0MW 121424047 EC50 = 9600 nM T69413 C2HV3U 134814234 EC50 = 5900 nM T69413 CYM2U5 134814235 EC50 = 14100 nM T69413 CDE3F4 134814236 EC50 = 9000 nM T69413 CGZ58C 134814237 EC50 = 3200 nM T69413 C8PK1D 134814239 EC50 = 11000 nM T69413 CHMF20 134814240 EC50 = 14500 nM T69413 CWO93M 134814241 EC50 = 1000 nM T69413 CSP5M8 134814242 EC50 = 2200 nM T69413 CY4I2L 134814243 EC50 = 8100 nM T69413 C4VMU5 134821714 EC50 = 1400 nM T69413 C9Z4KR 134821715 EC50 = 1600 nM T69413 CL7BV1 134821716 EC50 = 3100 nM T69413 C61MVQ 134821717 EC50 = 5900 nM T69413 C6XR3M 137322682 EC50 = 6400 nM T69413 C1N2LA 137322683 EC50 = 1800 nM T69413 C9ZV6G 142474254 EC50 = 6200 nM T69413 C6BL3M 142474259 EC50 > 100000 nM T69413 C47VHO 142474284 EC50 = 2000 nM T69413 CQ47VO 142474286 EC50 = 2500 nM T69413 CWP17Z 142474301 EC50 = 2500 nM T69413 C9HI0J 142474310 EC50 = 4200 nM T69413 CRAO80 142474312 EC50 = 7700 nM T69413 C3LI6V 142474314 EC50 > 100000 nM T69413 CXSW81 142474317 EC50 = 6600 nM T69413 CCOL46 142474341 EC50 = 1100 nM T69413 CEM34I 142474345 EC50 > 100000 nM T69413 CW8XZ7 142474362 EC50 = 2700 nM T69413 CW85FG 142474366 EC50 > 100000 nM T69413 C9VI0W 142474388 EC50 > 100000 nM T69413 CJIL08 145950108 EC50 = 6100 nM T69413 CCDO80 145950182 EC50 = 15900 nM T69413 CM5R1L 145950271 EC50 > 100000 nM T69413 C8QNS5 145950460 EC50 = 11200 nM T69413 C2I9BD 145950599 EC50 > 100000 nM T69413 C71PQJ 145950747 EC50 = 6700 nM T69413 C31HWR 145950974 EC50 = 800 nM T69413 COE96L 145951115 EC50 = 2900 nM T69413 C48CET 145951208 EC50 > 100000 nM T69413 C97MFE 145951513 EC50 = 7800 nM T69413 CUC0G3 145951548 EC50 = 13300 nM T69413 CB7M2W 145952689 EC50 > 100000 nM T69413 CK3MS4 145952954 EC50 = 15100 nM T69413 CNV89W 145953454 EC50 > 100000 nM T69413 CR0YL8 145953685 EC50 > 100000 nM T69413 C6ZN7V 145953743 EC50 > 100000 nM T69413 C9JA1R 145953899 EC50 > 100000 nM T69413 CQ13NI 145954809 EC50 = 800 nM T69413 CU8FL4 145957237 EC50 > 100000 nM T69413 C45MOE 145957733 EC50 > 100000 nM T69413 C0BQK1 145958763 EC50 = 14200 nM T69413 C4GBD8 145959032 EC50 = 4500 nM T69413 CJC80E 145959342 EC50 > 100000 nM T69413 C4YI0D 145959602 EC50 > 100000 nM T69413 C50IXS 145960575 EC50 = 8500 nM T69413 C7GYF3 145962934 EC50 = 37300 nM T69413 CK24RC 145963547 EC50 = 4400 nM T69413 CNVZ03 145963740 EC50 = 800 nM T69413 CDPB21 145963922 EC50 = 36600 nM T69413 CJ7P9Z 145963936 EC50 = 33200 nM T69413 CF9Q2E 145964087 EC50 = 8500 nM T69413 C0VPL9 145964186 EC50 = 24300 nM T69413 C4SMR3 145964356 EC50 = 8100 nM T69413 CC07PX 145964755 EC50 = 14000 nM T69413 C74WYJ 145964923 EC50 = 7800 nM T69413 CUEW50 145965845 EC50 = 2400 nM T69413 CB3QO7 145966464 EC50 = 8800 nM T69413 CWD97F 145967094 EC50 = 4100 nM T69413 C8WZJ7 145967208 EC50 = 1300 nM T69413 CONE49 145969362 EC50 = 14000 nM T69413 C2N4XU 145971371 EC50 = 11400 nM T69413 C4BW3T 145971431 EC50 = 10200 nM T69413 C32IBE 145971729 EC50 > 100000 nM T69413 CS2G6W 145971876 EC50 = 11700 nM T69413 CW3U1J 145971986 EC50 > 100000 nM T69413 CXYD94 145972055 EC50 = 6000 nM T69413 C4HO6U 145972098 EC50 = 5600 nM T69413 C92JRZ 145972340 EC50 = 3700 nM T69413 C75QVS 145972466 EC50 > 100000 nM T69413 CN9W1L 145972996 EC50 = 5900 nM T69413 CC7L0V 145974163 EC50 = 6600 nM T69413 CI9K7Q 145974183 EC50 = 37100 nM T69413 C5N6YS 145975456 EC50 = 19600 nM T69413 C34QUV 145975571 EC50 = 26000 nM T69413 C8TXH0 145975736 EC50 = 4400 nM T69413 C2Q3EB 145975788 EC50 = 1900 nM T69413 CN4ZD8 145976709 EC50 = 5900 nM T69413 C9UQB1 145977568 EC50 = 3000 nM T69413 CW2EH6 145977990 EC50 = 12400 nM T69413 C48OCG 145978477 EC50 = 5400 nM T69413 CB1DG9 145982662 EC50 > 100000 nM T69413 CB82EG 145983523 EC50 = 16300 nM T69413 CRG5N1 145983623 EC50 > 100000 nM T69413 CUH30J 145984027 EC50 > 100000 nM T69413 CR07ZJ 145984199 EC50 > 100000 nM T69413 CW50HZ 145984296 EC50 > 100000 nM T69413 C6M1PX 145984419 EC50 = 21900 nM T69413 C5NV0X 145984490 EC50 = 44200 nM T69413 C5I7KG 145984663 EC50 = 7100 nM T69413 CG2D8F 145985349 EC50 > 100000 nM T69413 C91PKE 145985504 EC50 = 3000 nM T69413 CH46SG 145985553 EC50 > 100000 nM T69413 C6GT9J 145985808 EC50 > 100000 nM T93145 D00YWP 9904 IC50 = 120000 nM T93145 D01FQV 517326 EC50 = 130000 nM T93145 D0X7HV 177852 EC50 = 8300 nM T93145 C38FDC 5729 IC50 = 32000 nM T93145 CHGI09 6597 IC50 > 2000000 nM T93145 CN65RY 62034 IC50 = 9500 nM T93145 CRJP61 443474 IC50 ~ 10000 nM T93145 CNP39D 6102761 EC50 = 57 nM T93145 CX8IJ9 9571025 IC50 = 5800 nM T93145 C9A1NJ 9799587 IC50 = 113 nM T93145 CI45SV 9886164 IC50 = 9300 nM T93145 C6M2XT 9909111 IC50 = 13 nM T93145 C1UE2K 9922541 IC50 = 51000 nM T93145 C0PQ1F 9948658 IC50 = 6400 nM T93145 CG5D7M 9995621 EC50 = 1400 nM T93145 CRKT64 10387163 IC50 = 55 nM T93145 C8LVC7 10500024 IC50 = 130 nM T93145 C4U9PR 10502897 IC50 = 4730 nM T93145 CA4IX5 10503143 IC50 = 20 nM T93145 CR17UB 10523081 IC50 = 87 nM T93145 C4UVJ5 10530132 IC50 = 110 nM T93145 C6Z5HJ 10544075 IC50 = 120 nM T93145 CL5IW7 10545701 IC50 = 98 nM T93145 CP5FB2 10547225 IC50 = 110 nM T93145 C6YSJ2 10547791 IC50 = 9300 nM T93145 C5PYM0 10551791 IC50 = 110 nM T93145 CG8RP7 10552429 IC50 = 1800 nM T93145 C8XL0B 10554131 IC50 = 130 nM T93145 CYT18D 10598084 IC50 = 32 nM T93145 CW2O6C 10600490 IC50 = 16 nM T93145 C6A8PO 10601861 IC50 = 380 nM T93145 C0W2NM 10620213 IC50 = 8 nM T93145 C1T8SC 10621272 IC50 = 29 nM T93145 C17BMI 10622643 IC50 = 19 nM T93145 CVGJ68 10643117 IC50 = 21 nM T93145 CBWA41 10643403 EC50 = 590 nM T93145 CST97A 10646927 IC50 = 8.4 nM T93145 C1R9CW 10665223 IC50 = 70 nM T93145 C51UJL 10672600 IC50 = 1300 nM T93145 CUXR17 10673527 IC50 = 230 nM T93145 CO9P3D 10681448 IC50 = 200000 nM T93145 CB40RK 10689528 IC50 = 6700 nM T93145 C6GF7L 10694289 IC50 = 140 nM T93145 CZ8LI0 10696482 IC50 = 73 nM T93145 CN46BQ 10706963 IC50 = 300 nM T93145 C6W4VU 10716132 IC50 = 61 nM T93145 CB1EY3 10719115 IC50 = 35 nM T93145 C2CZH5 10741908 IC50 = 920 nM T93145 C05NGP 10743090 IC50 = 15 nM T93145 CEP51A 10752088 IC50 = 35000 nM T93145 C4I3WK 10752484 IC50 = 6200 nM T93145 C0JQI7 10754328 IC50 = 9800 nM T93145 CL75FG 10759867 IC50 = 82 nM T93145 CQ89CI 10760269 IC50 = 77 nM T93145 CI7X3U 10784842 IC50 = 1490 nM T93145 C2WH0Z 10809954 IC50 = 47 nM T93145 C27EJT 10813807 IC50 = 10 nM T93145 C4IQ7K 10813808 IC50 = 66 nM T93145 C4T3SC 10834871 IC50 = 7.1 nM T93145 C30HDP 10836418 IC50 = 20 nM T93145 CP17LU 10838334 IC50 = 160 nM T93145 CIZ53L 10840047 IC50 = 77 nM T93145 CU0VY6 11726563 IC50 = 79 nM T93145 CB5K9D 14284032 IC50 = 36000 nM T93145 C14BEY 14786034 IC50 = 17300 nM T93145 C8W5UI 15482201 IC50 = 22600 nM T93145 CO6V7H 15482202 IC50 = 240 nM T93145 CD3I6X 21183546 IC50 = 9300 nM T93145 CH7RL6 21480124 IC50 = 203000 nM T93145 CL12AV 22287151 IC50 = 1500 nM T93145 CET87I 22287158 IC50 = 77 nM T93145 CL0O8G 22287173 IC50 = 2000 nM T93145 CDA20L 22287193 IC50 = 61500 nM T93145 CK9ES3 22287271 IC50 = 1200 nM T93145 C4A2GY 22287325 IC50 = 1000 nM T93145 CXD0T6 22287339 IC50 = 4150 nM T93145 CB83FT 22287432 IC50 = 2000 nM T93145 CZ9DO1 22287444 IC50 = 16100 nM T93145 CJ3B1I 23439395 IC50 = 300 nM T93145 CY59HW 23664150 IC50 = 34 nM T93145 C7IR9O 23667852 IC50 = 150 nM T93145 CS7F6M 23692717 IC50 = 140 nM T93145 C72HCA 44310889 IC50 = 5400 nM T93145 C51RDP 44311110 IC50 = 56000 nM T93145 COI68U 44311118 IC50 = 6700 nM T93145 CF2AL0 44311223 IC50 = 840 nM T93145 CD8P1W 44311845 IC50 = 3000 nM T93145 CFK74Q 44311863 IC50 = 150 nM T93145 CUPY94 44311864 IC50 = 16 nM T93145 CR02KV 44311903 IC50 = 560 nM T93145 CUZS09 44312004 IC50 = 16900 nM T93145 CH3S9T 44312015 IC50 = 42100 nM T93145 C4D6XM 44312040 IC50 = 2400 nM T93145 CYO78W 44312049 IC50 = 170000 nM T93145 CGB27I 44312050 IC50 = 21800 nM T93145 CT13KJ 44312051 IC50 = 47400 nM T93145 CW0TJ8 44312071 IC50 = 3660 nM T93145 CAI2C0 44312072 IC50 = 17700 nM T93145 C1QFP9 44312073 IC50 = 80000 nM T93145 CC1BQ7 44312074 IC50 = 219 nM T93145 C40PDZ 44312084 IC50 = 2800 nM T93145 CC8ZA5 44312085 IC50 = 145000 nM T93145 CDF38V 44312086 IC50 = 25000 nM T93145 C10PGI 44312087 IC50 = 380 nM T93145 CLRK42 44312120 IC50 = 596 nM T93145 C24LOX 44312151 IC50 = 30000 nM T93145 CY07TR 44312251 IC50 = 2700 nM T93145 CANO18 44312252 IC50 = 180 nM T93145 CD75HM 44312304 IC50 = 23 nM T93145 C1YO4K 44312327 IC50 = 126 nM T93145 CL30GX 44312331 IC50 = 22200 nM T93145 CE40IL 44312358 IC50 = 220000 nM T93145 CP6U1E 44312359 IC50 = 3800 nM T93145 C2QBW5 44312443 IC50 = 115 nM T93145 CE8W5C 44312513 IC50 = 60000 nM T93145 CTY4A8 44312541 IC50 > 3000 nM T93145 CWJ87R 44312558 IC50 = 45800 nM T93145 D0UQ6U 10569 IC50 = 20000 nM T43206 D02DGU 444795 IC50 = 199.53 nM T43206 D0D7CH 118622692 IC50 >= 30000 nM T43206 D0W1XE 91827457 IC50 > 10000 nM T43206 C25CAT 122184111 EC50 = 1600 nM T43206 CVS15Y 122184115 EC50 = 1900 nM T43206 C6R8ES 72721387 EC50 = 8360 nM T43206 CVEP92 91474 Ki = 12 nM T43206 CU8O6E 2360837 Ki = 220 nM T43206 C1LI3V 2855730 EC50 > 30000 nM T43206 CY0EV9 3399068 IC50 = 1680 nM T43206 C2J4CV 4158022 IC50 = 22600 nM T43206 C7CBK2 4170858 IC50 > 33000 nM T43206 CP4I7G 4289057 IC50 > 33000 nM T43206 CKCZ85 4396058 IC50 > 33000 nM T43206 C2ACB0 4419408 IC50 = 25000 nM T43206 CUT15M 4461168 IC50 = 30700 nM T43206 CUDT62 4597675 IC50 = 36500 nM T43206 C2ME9B 5079010 IC50 = 3220 nM T43206 C2LMW1 18565134 EC50 = 200 nM T43206 C0QKH8 18565138 EC50 = 86 nM T43206 CGS1R9 18565141 EC50 = 29 nM T43206 C4RYO8 19760309 IC50 > 10000 nM T43206 C38JEL 20704150 EC50 = 5000 nM T43206 C1FJU8 21824365 IC50 = 10200 nM T43206 CT3ZV5 23640021 IC50 = 21500 nM T43206 CF1S8P 25132150 IC50 > 20000 nM T43206 CNG1Z5 25132504 IC50 = 9900 nM T43206 CB56QH 25132505 IC50 > 20000 nM T43206 CS1EJ7 25234324 EC50 = 4200 nM T43206 CO1NQ0 41145803 IC50 > 5011.87 nM T43206 C9ZWM8 46866594 IC50 = 7200 nM T43206 CMR49F 46885348 IC50 > 20000 nM T43206 C18JYQ 46885349 IC50 = 10300 nM T43206 C4TLX3 46885390 IC50 = 17600 nM T43206 CSP3D8 46885467 IC50 = 9000 nM T43206 C8WM2R 46885468 IC50 = 16700 nM T43206 CP3O2L 46885469 IC50 > 20000 nM T43206 CG6JE7 46885508 IC50 = 11800 nM T43206 CX2U0L 46886033 IC50 > 20000 nM T43206 C6J5RT 46886034 IC50 = 7600 nM T43206 C2P5HX 54582225 IC50 = 7800 nM T43206 CQ02IF 54582227 IC50 > 10000 nM T43206 CS9O7F 54582228 IC50 = 5300 nM T43206 CPF9X2 54587076 IC50 = 9100 nM T43206 CFO23H 56837193 IC50 > 5011.87 nM T43206 CJ0I1V 71082496 IC50 = 10300 nM T43206 C1DR8E 71622396 EC50 = 2400 nM T43206 CK39WI 71816845 EC50 > 19000 nM T43206 CC8YU6 72720884 EC50 = 390 nM T43206 CMZ85K 72722807 EC50 = 7000 nM T43206 C2BQO3 72722945 EC50 = 6000 nM T43206 C6UWO5 74762670 EC50 = 4400 nM T43206 CJXG25 76284182 EC50 > 10000 nM T43206 C5PT4U 76314451 IC50 = 1300 nM T43206 CMW6O1 77620538 EC50 = 2800 nM T43206 C7ZMD9 78319220 IC50 = 5600 nM T43206 C4SA8H 86302482 EC50 > 10000 nM T43206 CBI06J 86346645 EC50 > 10000 nM T43206 C5VCM4 86690644 EC50 > 10000 nM T43206 CGFW70 86690646 EC50 > 10000 nM T43206 CNL0R1 87074581 IC50 = 110 nM T43206 C5MOV2 89659415 EC50 > 10000 nM T43206 CLW3O5 89665055 EC50 = 3800 nM T43206 C7E5RV 90200534 EC50 > 10000 nM T43206 CBCE70 90465832 IC50 > 30000 nM T43206 CEB82Q 90646513 IC50 > 30000 nM T43206 C0Z4BC 90646903 IC50 > 30000 nM T43206 C9FQ2N 90656122 IC50 = 13600 nM T43206 CF4M9V 90656123 IC50 = 12300 nM T43206 C5E6UV 90656124 IC50 = 10800 nM T43206 CS43BG 90656125 IC50 = 7600 nM T43206 C9TI2B 90656126 IC50 = 5500 nM T43206 C35ICO 90656127 IC50 = 6400 nM T43206 CI92WR 91664317 EC50 > 10000 nM T43206 C4S9EM 117964962 EC50 > 10000 nM T43206 CS4GJ9 117964973 EC50 > 10000 nM T43206 CDXK37 117964975 EC50 > 10000 nM T43206 CN6RT8 117964978 EC50 > 10000 nM T43206 C96BSK 117964998 EC50 > 10000 nM T43206 C56INY 118142016 IC50 > 30000 nM T43206 C79IOD 118207841 EC50 > 40000 nM T43206 C2FLM1 118207907 EC50 > 40000 nM T43206 CXW5M0 118207954 EC50 > 40000 nM T43206 C9UK5A 118207966 EC50 > 40000 nM T43206 C0PWH6 118207991 EC50 > 40000 nM T43206 C2U3TJ 118208018 EC50 > 40000 nM T43206 CZ2C3U 118208048 EC50 > 40000 nM T43206 C8N2PF 118208184 EC50 > 40000 nM T43206 C1ZRN9 118217594 EC50 > 40000 nM T43206 CAUT58 118217595 EC50 > 40000 nM T43206 CCK3J9 118217851 EC50 > 40000 nM T43206 CO5I3V 118217852 EC50 > 40000 nM T43206 CD5TJ3 118217853 EC50 > 40000 nM T43206 C6HSC3 118217854 EC50 > 40000 nM T43206 CEKH57 118217858 EC50 > 40000 nM T43206 C1CTB6 118217859 EC50 > 40000 nM T43206 C7U0XR 118217863 EC50 > 40000 nM T43206 CDP0H5 118217865 EC50 > 40000 nM T43206 C82YDU 118217866 EC50 > 40000 nM T43206 CQ60HK 118217867 EC50 > 40000 nM T43206 C9N7VY 118217868 EC50 > 40000 nM T43206 C6LC7H 118217869 EC50 > 40000 nM T43206 CV9G4S 118217870 EC50 > 40000 nM T43206 C8PR3G 118217871 EC50 > 40000 nM T43206 CZ3FX6 118217874 EC50 > 40000 nM T43206 CT0DV4 118217911 EC50 > 40000 nM T43206 C1QPW5 118217915 EC50 > 40000 nM T43206 C3YTM2 118217920 EC50 > 40000 nM T43206 CU0T7K 118217922 EC50 > 40000 nM T43206 C0ETA2 118217925 EC50 > 40000 nM T43206 C6X4IN 118217935 EC50 > 40000 nM T43206 CD01CA 118526849 EC50 = 8800 nM T43206 CBZ75K 118724654 EC50 > 7100 nM T43206 CB0AH7 118865631 IC50 > 30000 nM T43206 C27MYR 118865641 IC50 > 30000 nM T43206 C6TBD2 121345502 EC50 > 20000 nM T43206 C7D3AT 121429517 IC50 > 10000 nM T43206 C2JGN3 121429520 IC50 > 10000 nM T43206 CV5R4G 121470704 IC50 > 10000 nM T43206 CD89ZC 121480642 IC50 > 30000 nM T43206 CO6HF9 122180196 IC50 = 6200 nM T43206 CIX4M5 122180197 IC50 = 9400 nM T43206 CEW72J 122180199 IC50 = 7700 nM T43206 C5L1AS 122184114 EC50 = 2100 nM T43206 CL7EY2 122184139 EC50 = 9300 nM T43206 CE87BY 122184140 EC50 = 2200 nM T43206 CRY8N5 122190169 EC50 = 280 nM T43206 CB9GP5 122235238 IC50 > 10000 nM T43206 C0WAM1 122379290 EC50 = 5400 nM T43206 C4F9ZK 122669103 IC50 > 10000 nM T43206 CZH39M 122669106 IC50 > 10000 nM T43206 C0T8FO 122669173 IC50 > 10000 nM T43206 CD6X5P 122669265 EC50 > 10000 nM T43206 C0S7UB 122678562 IC50 > 10000 nM T43206 CY8S1P 122678563 IC50 > 10000 nM T43206 C0MUW2 122678576 IC50 > 10000 nM T43206 C2SQ9M 122678748 IC50 > 10000 nM T43206 CH1J6K 122678779 IC50 > 10000 nM T43206 CD9HN3 122678983 IC50 > 10000 nM T43206 CF39TE 122679031 IC50 > 10000 nM T43206 C0XWI7 127029952 IC50 > 30000 nM T43206 CD2LP9 130248006 IC50 = 7570 nM T43206 CXUK13 130261792 IC50 = 1740 nM T43206 CDV84X 131747741 EC50 > 20000 nM T43206 CP1U5T 134132295 IC50 > 10000 nM T43206 CX27TP 134693870 IC50 = 4113 nM T43206 CB3HG0 134817247 IC50 = 31622.78 nM T43206 C7MX4L 137633035 IC50 = 6000 nM T43206 CK1Z8N 137634168 IC50 = 30100 nM T43206 CLE56S 137636466 IC50 = 6800 nM T43206 CMT0R6 137637386 IC50 = 13000 nM T43206 CA1J8P 137639957 IC50 = 8000 nM T43206 CM6OP9 137640324 IC50 = 15000 nM T43206 CF3V7Z 137641972 IC50 = 8400 nM T43206 CHGQ98 137642611 IC50 = 9900 nM T43206 C9ZUD4 137644174 IC50 = 12500 nM T43206 C8HX6Q 137648178 IC50 = 7500 nM T43206 CLT70A 137654410 IC50 = 6800 nM T43206 C56NTF 137655509 IC50 = 6400 nM T43206 C9D2ME 137656123 IC50 = 26000 nM T43206 CM1L2U 137656343 IC50 = 11900 nM T43206 C0HPI9 137658927 IC50 = 5800 nM T43206 CK3X1N 137796283 IC50 > 10000 nM T43206 CM6OB9 138454290 IC50 = 501.19 nM T43206 CJ2R7W 141493565 EC50 > 10000 nM T43206 C7XT6D 141493567 EC50 > 10000 nM T43206 CC2BH9 145232219 IC50 > 10000 nM T43206 CDQK14 145954301 IC50 = 6200 nM T43206 C67MPG 145955616 IC50 > 33000 nM T43206 CR70ZO 145957041 IC50 = 600 nM T43206 C60CMX 145958026 IC50 > 33000 nM T43206 CL2HT7 145959111 IC50 = 9400 nM T43206 C4H9UY 145966156 EC50 > 2000 nM T43206 CB70AE 145980094 IC50 > 10000 nM T43206 C1JUC8 145982712 IC50 > 30000 nM T43206 C8G4QR 145982788 IC50 > 30000 nM T43206 CU0V8B 145984255 IC50 > 30000 nM T43206 CYRX35 145985210 IC50 > 30000 nM T43206 CP9Q8O 145985306 IC50 > 30000 nM T43206 CRTG03 145987785 IC50 > 10000 nM T43206 CC89OI 148034311 IC50 > 10000 nM T43206 CUFS62 155510496 EC50 = 6800 nM T43206 C9K7HE 155511006 IC50 > 31622.78 nM T43206 CE6V8Z 155511797 IC50 > 10000 nM T43206 CS93NA 155517530 IC50 > 31622.78 nM T43206 CE8R2A 155517869 IC50 > 31622.78 nM T43206 CU5Z8T 155522788 IC50 > 10000 nM T43206 C1DT9M 155525669 IC50 > 10000 nM T43206 C7Y5ZR 155526875 IC50 = 1995.26 nM T43206 CXS9T8 155526989 IC50 > 10000 nM T43206 C2HEC1 155530220 IC50 = 2511.89 nM T43206 CO9N5H 155530678 IC50 > 10000 nM T43206 CY0M8V 155532844 IC50 > 31622.78 nM T43206 CIUA10 155537856 IC50 > 10000 nM T43206 CLO98T 155539150 EC50 > 40000 nM T43206 COP7X8 155539171 IC50 > 10000 nM T43206 CMIT24 155542434 IC50 > 31622.78 nM T43206 C0V6EY 155543172 IC50 > 10000 nM T43206 CX7L0S 155544387 IC50 > 10000 nM T43206 CSK20E 155544524 IC50 > 10000 nM T43206 CYQ24A 155550306 IC50 > 31622.78 nM T43206 CF1D4A 155555172 IC50 = 1584.89 nM T43206 CBK1E5 155556708 IC50 > 10000 nM T43206 CQB48L 155556931 IC50 > 30000 nM T43206 C3FI7U 155560819 IC50 > 10000 nM T43206 CIBA72 155564665 IC50 > 30000 nM T43206 CA91EM 155564933 IC50 > 10000 nM T43206 CPF42S 155565257 IC50 > 10000 nM T43206 C6KMU5 122184108 EC50 = 1200 nM T43206 CV5CO0 122184112 EC50 = 1400 nM T43206 C63QAO 122184113 EC50 = 1100 nM T43206 CT3WD4 122184116 EC50 = 1500 nM T43206 CBHT23 122184117 EC50 = 2000 nM T43206 CH1EJ7 122184118 EC50 > 10000 nM T43206 C13QFC 122184133 EC50 = 1300 nM T43206 CO82BL 122184137 EC50 = 1800 nM T43206 CPM90L 122184138 EC50 = 9300 nM T43206 D0AJ5G 4076092 IC50 > 33000 nM T43206 D0B5FC 447912 Ki = 132 nM T43206 D0FB7S 473141 Ki = 12 nM T43206 D0K5QH 107722 Ki = 12 nM T43206 D0O1WJ 44241473 Ki = 172 nM T00442 D0J1VY 5281081 IC50 = 386 nM T00442 D0Y7PG 4659569 IC50 < 1 nM T00442 D01SGK 135565903 Ki = 1 nM T00442 D0E4WF 439176 Ki > 5400000 nM T00442 C1KG9Z 6792 IC50 = 6309.57 nM T00442 C7GLB3 2805447 Ki = 7900 nM T00442 CC4O6E 5152843 Ki = 251000 nM T00442 CLRD65 7147386 Ki = 6300 nM T00442 C0OE3C 10397916 IC50 = 18000 nM T00442 CF35YR 12468238 IC50 = 3400 nM T00442 C8C5OA 13130143 IC50 = 1700 nM T00442 CJLU70 14602319 IC50 > 10000 nM T00442 CK3C5U 15982971 Ki < 1 nM T00442 C3LM8W 19616700 Ki = 25000 nM T00442 C0I6QS 45266258 Ki = 5800000 nM T00442 C7Z3EI 45266259 Ki = 800000 nM T00442 CJO7Y5 45266260 Ki = 800000 nM T00442 CX5KA8 45266261 Ki = 6000000 nM T00442 C6OWN4 45266294 Ki = 500000 nM T00442 CSQW23 45588801 IC50 > 10000 nM T00442 C0OH4L 46865888 Ki = 17 nM T00442 C4JUD1 46865889 Ki = 1.6 nM T00442 CU9N6Q 46884860 Ki = 2.2 nM T00442 CE26QR 46884861 Ki = 9.2 nM T00442 CWF6J3 46884905 Ki = 1.3 nM T00442 CD8WZ0 46884906 Ki = 1.1 nM T00442 CE25JB 46884907 Ki = 10.2 nM T00442 CHI9F2 46884908 Ki = 17 nM T00442 CBZ6E7 46884909 Ki = 10.6 nM T00442 C6J5ZS 46884939 Ki = 16.6 nM T00442 C3FN6H 46884940 Ki = 6 nM T00442 CA03ZI 53379376 IC50 = 200 nM T00442 CVKW93 53379379 IC50 = 61 nM T00442 CNS4P0 53380912 IC50 = 47 nM T00442 CY7P2A 67405675 IC50 = 128 nM T00442 CJIM75 67418555 IC50 = 53 nM T00442 CGK4V8 67419355 IC50 = 87 nM T00442 CF80AB 67419505 IC50 = 3020 nM T00442 CBO31T 69929269 IC50 = 170 nM T00442 CHLG32 69931826 IC50 = 35 nM T00442 C5FVM1 69932256 IC50 = 706 nM T00442 CEDU65 69932313 IC50 = 680 nM T00442 C0W4YT 69932481 IC50 = 101 nM T00442 C9I8JN 69932517 IC50 = 1500 nM T00442 CXO59G 69932543 IC50 > 5000 nM T00442 C6C3SV 69932581 IC50 = 2400 nM T00442 C0WFN4 71395955 IC50 = 19.95 nM T00442 CMA72V 89466901 IC50 = 84 nM T00442 CQG3M5 89467005 IC50 = 55 nM T00442 CO1F2M 118736597 IC50 = 400 nM T00442 CVD30G 118736600 IC50 > 10000 nM T00442 CFCS69 118736601 IC50 = 4500 nM T00442 C8CNJ1 118736602 IC50 = 5800 nM T00442 C5SB8X 118736603 IC50 = 5500 nM T00442 C0FIS1 118736604 IC50 = 160 nM T00442 CJCQ91 118736605 IC50 = 140 nM T00442 CZ1FH9 118736606 IC50 = 140 nM T00442 CM2T4P 118736607 IC50 = 88 nM T00442 CBLT83 118736608 IC50 = 57 nM T00442 CDZ9V5 118736609 IC50 = 1900 nM T00442 CZ85HC 118736610 IC50 = 13000 nM T00442 CF0Z7Q 122439995 IC50 = 1.995 nM T00442 C1PE9K 122440001 IC50 = 3.981 nM T00442 CQ9FG1 122440007 IC50 = 199.53 nM T00442 CRV7L1 122440022 IC50 = 10 nM T00442 C9TP2N 122440029 IC50 = 19.95 nM T00442 CKS61V 122440030 IC50 = 79.43 nM T00442 CB54TV 122440031 IC50 = 7.943 nM T00442 C5R2JV 122441915 IC50 = 6.31 nM T00442 C4OJ6D 122441945 IC50 = 316.23 nM T00442 C6NL1P 122441948 IC50 > 10000 nM T00442 C7A5TQ 122441954 IC50 = 1584.89 nM T00442 CI65KH 122441965 IC50 = 6.31 nM T00442 CPLQ64 122441976 IC50 = 63.1 nM T00442 C85YVR 122441981 IC50 = 1258.93 nM T00442 C92VAF 122442004 IC50 = 19.95 nM T00442 C36XNY 122442007 IC50 = 3.162 nM T00442 C4WVK0 122442029 IC50 = 3.981 nM T00442 CD9IE5 122442045 IC50 > 10000 nM T00442 CA35KX 122442051 IC50 = 1.995 nM T00442 C7KTJ8 127046300 IC50 = 456 nM T00442 CJ6WA2 127046783 IC50 > 5000 nM T00442 C0ZWY6 127047871 IC50 = 962 nM T00442 CB5I2N 127047926 IC50 = 1667 nM T00442 CQU46R 127048055 IC50 = 826 nM T00442 C8F2XG 127048056 IC50 = 672 nM T00442 C7VJ3D 127048057 IC50 = 574 nM T00442 C8DT5E 127048058 IC50 = 49.5 nM T00442 C0OY3S 127050334 IC50 = 179 nM T00442 CTH9J4 127050335 IC50 = 54 nM T00442 CQA4M8 127050621 IC50 = 648 nM T00442 CK0DI2 129165296 IC50 = 50 nM T00442 C83LIY 129165316 IC50 = 10 nM T00442 C8BOL3 129165356 IC50 = 10 nM T00442 CFGM98 129165376 IC50 = 220 nM T00442 C3H8LN 129165377 IC50 = 60 nM T00442 CF67NH 129165444 IC50 = 630 nM T00442 CG3OP9 129165448 IC50 = 63 nM T00442 CJGE94 129165458 IC50 = 40 nM T00442 CDT58P 129165460 IC50 = 16 nM T00442 C0F7CK 129165469 IC50 = 400 nM T00442 CHZ7N2 129165491 IC50 = 250 nM T00442 CXU3W9 129165493 IC50 = 6.3 nM T00442 CJ51DV 129165494 IC50 = 38 nM T00442 CY5X3U 129165527 IC50 = 100 nM T00442 CI0C1P 129165534 IC50 = 13 nM T00442 C1DPO0 129165543 IC50 = 40 nM T00442 CTUA67 129165554 IC50 = 50 nM T00442 CO0VS6 129165556 IC50 = 40 nM T00442 CW2S3J 129165564 IC50 = 450 nM T00442 C8OC4X 136934927 IC50 = 2100 nM T00442 CK0ZP6 140931610 IC50 = 6300 nM T00442 C48UMS 145949230 IC50 = 1584.89 nM T00442 CD3M0U 145950392 IC50 > 10000 nM T00442 CVR04X 145951510 IC50 = 251.19 nM T00442 C7SMJ2 145956792 IC50 = 3981.07 nM T00442 CHO0E4 155518634 IC50 = 1600 nM T00442 C6ATD2 155523978 IC50 = 2000 nM T00442 C3B0SN 155543374 IC50 > 10000 nM T00442 CCNW79 155543901 IC50 = 2000 nM T00442 CQLM48 155562927 IC50 > 10000 nM T00442 D0FO2B 1923 IC50 = 3162.28 nM T08985 D0F8UV 9941306 IC50 = 33.27 nM T08985 CQV8M4 444296 IC50 = 11.99 nM T08985 CV4A7J 444317 IC50 = 13 nM T08985 C72HYA 657089 IC50 = 112.98 nM T08985 CEUF82 657090 IC50 = 19.1 nM T08985 C9RY6N 9811991 IC50 = 100 nM T08985 CL4DJ6 9832889 IC50 = 214.78 nM T08985 CW10FH 9833347 IC50 = 20.8 nM T08985 CUWO10 9876066 IC50 = 193.2 nM T08985 CCZ01N 9897305 IC50 = 262.42 nM T08985 CB3IG9 9897777 IC50 = 381.07 nM T08985 CZU78V 9897907 IC50 = 74.64 nM T08985 CTXH45 9919490 IC50 = 45.5 nM T08985 CHK1Z8 9963312 IC50 = 147.23 nM T08985 C4Z0FA 9963581 IC50 = 35.97 nM T08985 C1E5OU 10123773 IC50 = 27.99 nM T08985 CUR10K 10124095 IC50 = 161.06 nM T08985 C30DLM 10124164 IC50 = 8.851 nM T08985 CMS47O 10124254 IC50 = 333.43 nM T08985 CR2PU7 10124289 IC50 = 2.198 nM T08985 C2FM6I 10148151 IC50 = 39.99 nM T08985 C7SU2D 10148210 IC50 = 462.38 nM T08985 CF1MU7 10148239 IC50 = 238.23 nM T08985 CNZK76 10170210 IC50 = 147.23 nM T08985 CC12RO 10170463 IC50 = 328.1 nM T08985 CQ54TI 10170557 IC50 = 8.954 nM T08985 C27VQZ 10197428 IC50 = 164.06 nM T08985 CM6BG4 10213994 IC50 = 11.09 nM T08985 CA1NZ7 10235097 IC50 = 416.87 nM T08985 C3WYU0 10235345 IC50 = 26 nM T08985 C7LG2E 10240569 IC50 = 4.498 nM T08985 CV1B6M 10306569 IC50 = 7.998 nM T08985 C54CNY 10312856 IC50 = 1438.8 nM T08985 CNZ8X9 10312910 IC50 = 16.98 nM T08985 CI1V0O 10418684 IC50 = 1.698 nM T08985 CKR98M 11170737 IC50 = 187.93 nM T08985 CKQ27V 11766591 IC50 = 2 nM T08985 CHOS82 15605382 IC50 = 1000 nM T08985 CXCT75 15605520 IC50 = 14.29 nM T08985 C7KJG8 16039076 IC50 = 3.999 nM T08985 C7T9PO 16200121 IC50 = 15 nM T08985 CW5Q9I 24853157 IC50 = 3.304 nM T08985 CATI05 25183240 IC50 = 7.096 nM T08985 C3D0SU 44345246 IC50 = 7.499 nM T08985 C0XN8P 44345247 IC50 = 95.5 nM T08985 CWC93Q 44345248 IC50 = 103.99 nM T08985 C5BD0I 44345270 IC50 = 11.51 nM T08985 C3J6CN 44345379 IC50 = 8.892 nM T08985 CWSM24 44345380 IC50 = 39.99 nM T08985 CLU4S7 44345392 IC50 = 153.11 nM T08985 C34HUZ 44345422 IC50 = 41.4 nM T08985 C5LY1X 44345423 IC50 = 7144.96 nM T08985 CZX8Q5 44345424 IC50 = 7144.96 nM T08985 CB09DO 44345425 IC50 = 65.01 nM T08985 C7SZ3I 44345427 IC50 = 5.794 nM T08985 CN1V4P 44345443 IC50 = 161.06 nM T08985 CR5Q7D 44345444 IC50 = 76.91 nM T08985 C70SHG 44345445 IC50 = 85.9 nM T08985 C2QUZ8 44345446 IC50 = 87.5 nM T08985 CUE23S 44345466 IC50 = 229.61 nM T08985 CZE64Q 44345467 IC50 = 11.99 nM T08985 CR84CY 44345474 IC50 = 61.38 nM T08985 C0O2WZ 44345475 IC50 = 66.22 nM T08985 CR70WK 44345495 IC50 = 126.47 nM T08985 CUP1I6 44345496 IC50 = 130.02 nM T08985 CPQ18E 44345505 IC50 = 1819.7 nM T08985 CJ9KM8 44345506 IC50 = 2630.27 nM T08985 CSRL31 44345507 IC50 = 3155 nM T08985 CN71VA 44345508 IC50 = 666.81 nM T08985 CK8M0N 44345509 IC50 = 716.14 nM T08985 CW6PD3 44345523 IC50 = 66.99 nM T08985 C93SHE 44345524 IC50 = 69.34 nM T08985 CVG6N2 44345542 IC50 = 277.97 nM T08985 C7MYJ9 44345543 IC50 = 3572.73 nM T08985 C5T1SH 44345544 IC50 = 4549.88 nM T08985 C63INV 44345545 IC50 = 5000.35 nM T08985 CWMN10 44345567 IC50 = 666.81 nM T08985 CD5ZM2 44345568 IC50 = 676.08 nM T08985 CL0O5G 44345569 IC50 = 207.97 nM T08985 CY3T4U 44345577 IC50 = 847.23 nM T08985 CN2Y0Z 44345578 IC50 = 1000 nM T08985 C9UV4S 44345579 IC50 = 1352.07 nM T08985 CMJX47 44345580 IC50 = 44.98 nM T08985 CEUV78 44345593 IC50 = 142.89 nM T08985 C5R2KL 44345594 IC50 = 73.96 nM T08985 C1WI4B 44345595 IC50 = 76.03 nM T08985 CD7T9I 44345603 IC50 = 100 nM T08985 C91WIJ 44345604 IC50 = 100.93 nM T08985 C9FMV4 44345605 IC50 = 133.35 nM T08985 CK0ZG8 44345614 IC50 = 14.29 nM T08985 CAN1Y6 44345615 IC50 = 15.21 nM T08985 CK53PQ 44345653 IC50 = 46.99 nM T08985 CH7BV1 44345670 IC50 = 308.32 nM T08985 C9BR8C 44345671 IC50 = 384.59 nM T08985 C2F7PI 44345672 IC50 = 416.87 nM T08985 CIL0O2 44345673 IC50 = 454.99 nM T08985 CB65VE 44345674 IC50 = 26 nM T08985 CO2WK3 44345682 IC50 = 636.8 nM T08985 CH4V2Y 44345683 IC50 = 111.17 nM T08985 C7KM2N 44345684 IC50 = 112.98 nM T08985 CC4DA5 44345685 IC50 = 48.98 nM T08985 CE13QH 44345704 IC50 = 34.43 nM T08985 CH7N6O 44345705 IC50 = 39.99 nM T08985 CQ36UK 44345721 IC50 = 217.27 nM T08985 C6MC9V 44345722 IC50 = 333.43 nM T08985 C01LEO 44345723 IC50 = 16.9 nM T08985 C2GBY7 44345724 IC50 = 20 nM T08985 CNW17O 44345725 IC50 = 22.8 nM T08985 C5V3TD 44345749 IC50 = 500.03 nM T08985 C9PE3D 44345769 IC50 = 615.18 nM T08985 C07NTD 44345770 IC50 = 39.99 nM T08985 CMUW62 44345771 IC50 = 29.38 nM T08985 C4VQ2F 44345772 IC50 = 45.5 nM T08985 C5Q6ED 44345785 IC50 = 1614.36 nM T08985 C20TRL 44345786 IC50 = 2630.27 nM T08985 CB25HM 44345808 IC50 = 1315.22 nM T08985 CUX1P2 44345809 IC50 = 1352.07 nM T08985 C39JSZ 44345824 IC50 = 399.94 nM T08985 C9SIB6 44345837 IC50 = 4168.69 nM T08985 CC0S3G 44345880 IC50 = 159.96 nM T08985 C9H2NR 44345881 IC50 = 130.02 nM T08985 C82KYS 44345884 IC50 = 827.94 nM T08985 CO57SG 44345885 IC50 = 944.06 nM T08985 CA14XC 44345901 IC50 = 21.98 nM T08985 CF7TC1 44345902 IC50 = 22.7 nM T08985 C6UKZ8 44345904 IC50 = 50 nM T08985 CCP34F 44345905 IC50 = 56.49 nM T08985 C25PSO 44345906 IC50 = 207.97 nM T08985 CQLB39 44345916 IC50 = 238.23 nM T08985 CJ0HV2 44345917 IC50 = 319.89 nM T08985 CK7NO8 44345941 IC50 = 3.199 nM T08985 C29UEO 44345942 IC50 = 4.295 nM T08985 CEW78H 44345943 IC50 = 5.794 nM T08985 C6JKQ5 44345969 IC50 = 2.301 nM T08985 CM1U8V 44345970 IC50 = 3.199 nM T08985 C8R0ZL 44345972 IC50 = 33.11 nM T08985 C70ROP 44345985 IC50 = 238.23 nM T08985 CA0TC5 44345986 IC50 = 263.03 nM T08985 CG7NR8 44345996 IC50 = 7.499 nM T08985 C25XGC 44346014 IC50 = 26 nM T08985 CBZT63 44346015 IC50 = 17.22 nM T08985 C1K9XZ 44346016 IC50 = 20 nM T08985 CVI7B8 44346024 IC50 = 16 nM T08985 C0PGT3 44346029 IC50 = 4549.88 nM T08985 CG10JK 44346030 IC50 = 5000.35 nM T08985 CKD34G 44346031 IC50 = 4.898 nM T08985 CXU90M 44346032 IC50 = 9.29 nM T08985 CRHF21 44346033 IC50 = 10 nM T08985 C3S5DT 44346035 IC50 = 11.51 nM T08985 C3YZ4X 44346036 IC50 = 11.69 nM T08985 C47FDJ 71457972 IC50 = 381.07 nM T20178 D09QEI 4740 IC50 = 85000 nM T20178 D0C4YC 4075 IC50 = 20600000 nM T20178 D05VZE 119031 IC50 = 1001 nM T20178 D0T5PO 5092 IC50 = 200 nM T20178 D07FHZ 5087 IC50 = 50000 nM T20178 D0T3ME 156422 EC50 = 18 nM T20178 CY9A0M 66065 IC50 = 12500 nM T20178 C21OTL 151419 IC50 > 200000 nM T20178 CQDJ34 428211 IC50 > 100000 nM T20178 CPE2J7 461663 IC50 = 12000 nM T20178 CNH7C2 461664 IC50 = 2900 nM T20178 C13KWU 461665 IC50 = 260000 nM T20178 C8PR3E 461666 IC50 = 380 nM T20178 CS3J5K 467265 IC50 = 400 nM T20178 C9YR0M 676987 IC50 = 200000 nM T20178 CZ37KX 874861 IC50 > 100000 nM T20178 CW9TZ3 1137620 IC50 > 100000 nM T20178 CDQ2E4 1367407 IC50 = 42300 nM T20178 C6O7AP 1582566 IC50 = 14000 nM T20178 C5CW1K 3081830 IC50 > 200000 nM T20178 CE80AQ 5327044 IC50 = 22000 nM T20178 CI13SQ 6523638 IC50 = 5750 nM T20178 C32HOB 9797095 IC50 = 150000 nM T20178 C2EV5L 9824551 IC50 = 10000 nM T20178 CJQ20V 9840218 IC50 = 120000 nM T20178 CF5T8E 9840925 IC50 = 7500 nM T20178 CF7AS4 9841064 IC50 = 51000 nM T20178 CX35SG 9850770 EC50 = 50 nM T20178 C34KGT 9892658 EC50 = 9 nM T20178 C13TVP 9904193 IC50 = 6000 nM T20178 CF1OJ6 9907022 IC50 = 70000 nM T20178 C49ILA 9936768 EC50 = 19 nM T20178 C2KI0C 9948975 IC50 = 3000 nM T20178 CFDN06 9949152 IC50 = 62000 nM T20178 C6XV8K 10019033 IC50 = 5000 nM T20178 C1NSK8 10091288 IC50 = 5600 nM T20178 CK5CJ9 10165915 EC50 = 42 nM T20178 CCE2T5 10229750 EC50 = 20 nM T20178 CBCW38 10256389 EC50 = 9 nM T20178 CV1WZ5 10301047 EC50 = 36 nM T20178 C1QM5I 10360825 IC50 = 60000 nM T20178 C4FOR3 10423517 IC50 = 4000 nM T20178 CL7N3F 10452587 IC50 = 450 nM T20178 CK3CH6 10498658 IC50 = 37000 nM T20178 C1BNW9 10498936 IC50 > 25000 nM T20178 CMTG10 10500152 IC50 > 100000 nM T20178 C1X5GM 10503011 IC50 = 11000 nM T20178 C49VUL 10515426 IC50 = 5000 nM T20178 CYH81M 10515726 IC50 > 200000 nM T20178 C3WQD5 10520713 IC50 = 15000 nM T20178 CZ8Y2I 10522445 IC50 = 38000 nM T20178 CY1V5H 10522585 IC50 = 15000 nM T20178 C63OLU 10527621 IC50 > 50000 nM T20178 C3S8WZ 10538504 IC50 = 55000 nM T20178 CI3GV1 10539258 IC50 > 25000 nM T20178 CN97DW 10539960 IC50 > 200000 nM T20178 C1HP3M 10541869 IC50 > 25000 nM T20178 CAKR74 10543322 IC50 = 35000 nM T20178 C2E0DT 10546983 IC50 = 175000 nM T20178 CB4QK3 10547110 IC50 = 1000 nM T20178 C7V5IZ 10547590 IC50 > 100000 nM T20178 CIZ1H6 10548866 IC50 = 51000 nM T20178 CRZ8G2 10553070 IC50 > 25000 nM T20178 C08KTS 10570106 IC50 = 39000 nM T20178 CWH0D5 10570570 IC50 = 14000 nM T20178 C3KPO8 10571036 IC50 = 12000 nM T20178 CE4N3P 10572133 IC50 = 15000 nM T20178 C7AHE4 10573618 IC50 = 55000 nM T20178 C8QJH2 10590173 IC50 = 25000 nM T20178 C0YCK7 10591397 IC50 = 33000 nM T20178 CRB09M 10594315 IC50 = 68000 nM T20178 CR0B3N 10595485 IC50 = 60000 nM T20178 C7XQS9 10613843 IC50 > 25000 nM T20178 C12ZAL 10619896 IC50 = 53000 nM T20178 C4XID0 10636108 IC50 = 9000 nM T20178 CKOB90 10639329 IC50 = 5000 nM T20178 C0KFZ3 10640389 IC50 = 21000 nM T20178 C0WS8E 10660380 IC50 = 10000 nM T20178 C3KHD5 10661296 IC50 > 200000 nM T20178 C8UN3P 10663883 IC50 = 100000 nM T20178 CHD97W 10665860 IC50 = 48000 nM T20178 CK0BJ2 10669458 IC50 = 34000 nM T20178 C0PXG8 10683932 IC50 = 10000 nM T20178 C7RK6Y 10685254 IC50 > 25000 nM T20178 C5UIP8 10685991 IC50 > 25000 nM T20178 CW4V3K 10686085 IC50 = 9000 nM T20178 C0S1YO 10687089 IC50 = 89000 nM T20178 CQ5BS6 10688147 IC50 = 20000 nM T20178 CH29QB 10688432 IC50 > 25000 nM T20178 C61YEC 10690566 IC50 = 37000 nM T20178 CZ6S3J 10692755 IC50 > 200000 nM T20178 C49ACR 10694297 IC50 = 13000 nM T20178 CY1JS2 10694592 IC50 = 84000 nM T20178 CFB7U5 10708682 IC50 = 2000 nM T20178 C1GE5N 10712721 IC50 = 16000 nM T20178 C3A9FI 10713603 IC50 > 25000 nM T20178 CVP4S5 10713794 IC50 = 35000 nM T20178 CXP38D 10730172 IC50 > 200000 nM T20178 CEA8F4 10731271 IC50 > 25000 nM T20178 C3EWQ9 10731615 IC50 = 75000 nM T20178 CWS49T 10732591 IC50 > 25000 nM T20178 C5IO6M 10733368 IC50 = 50000 nM T20178 CQ5FM6 10734444 IC50 = 3000 nM T20178 CMN70S 10735519 IC50 = 15000 nM T20178 CWX49K 10736217 IC50 = 5000 nM T20178 C3UG9F 10736883 IC50 = 22000 nM T20178 C1BJ5K 10737740 IC50 > 200000 nM T20178 CRO94K 10740359 IC50 > 25000 nM T20178 CIRT20 10755908 IC50 = 55000 nM T20178 CK2X0E 10756895 IC50 > 100000 nM T20178 C0NL2W 10758494 IC50 = 18000 nM T20178 CTV0Z7 10759371 IC50 = 20000 nM T20178 C71RHU 10762006 IC50 = 9000 nM T20178 C6OD5G 10764262 IC50 = 64000 nM T20178 CKT0A9 10765443 IC50 = 7900 nM T20178 CGVQ48 10779971 IC50 = 12000 nM T20178 C5KY6T 10780887 IC50 > 25000 nM T20178 C41JMB 10782487 IC50 > 200000 nM T20178 CAY0N3 10787769 IC50 > 25000 nM T20178 C28QZK 10803497 IC50 > 100000 nM T20178 CL6RT8 10806631 IC50 = 6000 nM T20178 C3PE6Z 10808807 IC50 = 11000 nM T20178 C1ZOT3 10812014 IC50 = 4700 nM T20178 CM98RG 10826387 IC50 = 5000 nM T20178 CV8SL6 10827468 IC50 = 48000 nM T20178 C2I8UZ 10831571 IC50 = 13000 nM T20178 C5XT1B 10831577 IC50 = 130000 nM T20178 C4Z1VG 10836140 IC50 = 4200 nM T20178 C60MTS 10838771 IC50 > 50000 nM T20178 CZ6AO2 10850191 IC50 > 25000 nM T20178 CQ84TR 10852312 IC50 = 11000 nM T20178 CXT17W 10854252 IC50 > 25000 nM T20178 C7E0YH 10896702 EC50 = 11 nM T20178 CXY64V 11731370 EC50 = 16 nM T20178 C04DFH 11783486 IC50 = 928 nM T20178 C28RVB 11792503 IC50 > 100000 nM T20178 C3VO5H 11824148 IC50 = 1606 nM T20178 CM52YU 14422379 IC50 = 28000 nM T20178 C8USX1 25118615 IC50 = 10000 nM T20178 C94PAD 44382351 IC50 = 25000 nM T20178 CA42ZX 44382442 IC50 > 200000 nM T20178 C8ACR4 44382640 IC50 = 50000 nM T20178 CBI2Y3 44383341 IC50 = 19000 nM T20178 CZB81D 44395506 IC50 = 10.4 nM T20178 CN6E2O 45265215 IC50 = 20000 nM T20178 CBH42D 118711553 IC50 = 20300 nM T20178 C5O8KD 124222736 IC50 = 1200 nM T20178 CE05SO 127038031 IC50 = 15000 nM T20178 C0TOH8 127038032 IC50 = 20000 nM T20178 C70RME 127038387 IC50 = 20000 nM T20178 C2GP1N 127038388 IC50 = 20000 nM T20178 CK5VZ6 127038389 IC50 = 20000 nM T20178 C4G5DV 127038390 IC50 = 20000 nM T20178 C92ENQ 127038391 IC50 = 20000 nM T20178 C0IPO4 127038747 IC50 = 30000 nM T20178 C3CI0D 127038748 IC50 = 30000 nM T20178 C3WCF7 127038749 IC50 = 20000 nM T20178 CS92HL 127039093 IC50 = 40000 nM T20178 C50OZL 127039403 IC50 = 15000 nM T20178 CX14NZ 127041410 IC50 = 10000 nM T20178 C2YG4X 127041411 IC50 > 60000 nM T20178 CW1ZD3 127041716 IC50 = 10000 nM T20178 CEDC62 127041718 IC50 = 20000 nM T20178 CD09BY 127050135 IC50 = 32600 nM T20178 CF2GT1 127051022 IC50 = 20700 nM T20178 CLD3J6 139562057 IC50 = 290 nM T20178 CY95MV 145948918 IC50 = 11900 nM T20178 CN54LI 145960710 IC50 = 2250 nM T20178 CYZW31 145961618 IC50 = 1990 nM T20178 CO5WL0 145961950 IC50 = 2710 nM T20178 C27UMT 145962409 IC50 = 2130 nM T20178 C0UG8V 145962807 IC50 = 4800 nM T20178 CW1OQ2 145963071 IC50 = 2140 nM T20178 C18ECW 145964594 IC50 = 11000 nM T20178 C4VHJ3 145964847 IC50 > 30000 nM T20178 CNT8P1 145965028 IC50 = 6000 nM T20178 CCMN84 145965066 IC50 > 30000 nM T20178 CO4T0U 145965354 IC50 = 9000 nM T20178 CR3YI7 145966075 IC50 = 20000 nM T20178 CFVT97 145966246 IC50 = 30000 nM T20178 CO43ZI 145966328 IC50 = 11000 nM T20178 CQD30F 145966692 IC50 = 20000 nM T20178 C2MEV8 145966854 IC50 = 4000 nM T20178 CI2B6G 145967228 IC50 = 18000 nM T20178 CJDX46 145967246 IC50 = 15000 nM T20178 C98KUB 145967291 IC50 = 20000 nM T20178 CW06TA 145967459 IC50 = 6000 nM T20178 C6L5WA 145969826 IC50 > 30000 nM T20178 C0C6FU 145971874 IC50 = 12000 nM T20178 CKME54 145972363 IC50 = 12000 nM T20178 C0WT5G 145972831 IC50 = 4000 nM T20178 C9PS6E 145973432 IC50 = 300 nM T20178 C9Y2GW 145973540 IC50 = 15000 nM T20178 CWMO63 145974409 IC50 = 500 nM T20178 CP7JG6 145974587 IC50 > 30000 nM T20178 C0A9IQ 145974635 IC50 > 30000 nM T20178 CB84OT 145974761 IC50 > 30000 nM T20178 C8LSE1 145974997 IC50 > 30000 nM T20178 CG0X5M 145976094 IC50 = 11000 nM T20178 CIXO30 145976316 IC50 > 30000 nM T20178 C4VKS2 145976571 IC50 > 30000 nM T20178 CD7KG0 145976625 IC50 > 30000 nM T20178 C0QWS3 145976834 IC50 = 4000 nM T20178 CQ1X3N 145977395 IC50 = 4000 nM T20178 C4B1OR 145977408 IC50 = 7000 nM T20178 CW5E2K 145977530 IC50 = 25000 nM T20178 CHR1E5 145977810 IC50 = 28000 nM T20178 CXR3U7 145977818 IC50 > 30000 nM T20178 CI73TP 145977952 IC50 = 30000 nM T20178 CQN5R6 145977985 IC50 = 8000 nM T20178 C3HUA7 145978193 IC50 = 28000 nM T20178 CP0AQ4 145978399 IC50 = 30000 nM T20178 CHOY97 145978512 IC50 > 30000 nM T20178 CQAY27 145981693 IC50 = 540 nM T20178 CH62WV 145985146 IC50 = 360 nM T20178 D02UYR 9907830 IC50 = 269 nM T20178 D0H2PA 9886977 IC50 = 48 nM T87749 CRS87L 118732224 IC50 = 4100 nM T87749 CSD16Y 118732229 IC50 = 3560 nM T87749 C9E3GH 134137378 IC50 = 1190 nM T87749 CP8I7R 137634541 IC50 = 320 nM T87749 C7SU2J 155519745 IC50 = 130 nM T87749 CQ4JP9 155540392 IC50 = 260 nM T58924 D0E3TC 44259 IC50 = 227 nM T58924 CV63UL 67240318 IC50 > 10000 nM T58924 C2AN7T 134611886 IC50 > 100000 nM T58924 C2MD1Q 155513187 IC50 > 10000 nM T00890 D0N0ES 938 EC50 > 10000 nM T00890 D01DDN 56950369 EC50 = 96 nM T00890 D0K1HO 51576 EC50 = 316 nM T00890 C2SZP8 99209 EC50 < 10000 nM T00890 C9HSZ4 283475 EC50 = 1905.46 nM T00890 CE5F8B 653819 EC50 = 5888.44 nM T00890 CWV37H 1447952 EC50 = 389.05 nM T00890 CJX8T7 2103992 EC50 = 891.25 nM T00890 C7UI0X 2771812 EC50 = 3235.94 nM T00890 CWY8I2 2776549 EC50 = 1995.26 nM T00890 CU62TL 2829816 EC50 = 158.49 nM T00890 CP9Z1W 2833647 EC50 = 630.96 nM T00890 CGD5M8 2942936 EC50 = 309.03 nM T00890 C0BER5 3671930 EC50 < 10000 nM T00890 CW36OS 3684804 EC50 = 2041.74 nM T00890 CFP65N 3729086 EC50 = 229.09 nM T00890 CP35CQ 3824366 EC50 = 2454.71 nM T00890 CAGJ29 4712703 EC50 = 3388.44 nM T00890 CQ2IY4 4738197 EC50 = 588.84 nM T00890 CDW7B3 4992776 EC50 = 309.03 nM T00890 CES08X 9971057 EC50 = 5011.87 nM T00890 CCUP10 10013684 EC50 = 331.13 nM T00890 CAYF98 10014206 EC50 = 288.4 nM T00890 CIPD39 10058774 EC50 = 7413.1 nM T00890 C5SB2K 10198518 EC50 = 1096.48 nM T00890 CWX34V 10263467 EC50 = 199.53 nM T00890 CSY4E7 10330955 EC50 = 3090.3 nM T00890 CF41BU 10331019 EC50 = 691.83 nM T00890 CZ01LF 10353934 EC50 = 3019.95 nM T00890 CYDU34 10398515 EC50 = 257.04 nM T00890 C0XQ3T 10398583 EC50 = 316.23 nM T00890 C5W8ZT 10421571 EC50 = 257.04 nM T00890 CRUE32 10422270 EC50 = 302 nM T00890 CG95LV 10446870 EC50 < 10000 nM T00890 C6TNZ8 10449244 EC50 < 10000 nM T00890 C4P5OW 10465474 EC50 = 2344.23 nM T00890 CXG5D6 11183678 EC50 = 4200 nM T00890 CX3R0C 11184165 EC50 = 6200 nM T00890 C7T5ZM 11218626 EC50 = 1800 nM T00890 CE9H6X 11219885 EC50 = 12600 nM T00890 CSHA60 11264843 EC50 = 9900 nM T00890 C1PO6Q 11276453 EC50 = 270 nM T00890 C6F1PI 11311474 EC50 = 3700 nM T00890 C2DAT1 11322738 EC50 = 22000 nM T00890 C4L1NT 11322761 EC50 = 24000 nM T00890 CG6T1I 11322762 EC50 = 36000 nM T00890 CYA94T 11324121 EC50 = 4100 nM T00890 CG2T6U 11379903 EC50 = 690 nM T00890 CM25BS 11380943 EC50 = 4900 nM T00890 C2W9MS 11413114 EC50 = 5100 nM T00890 C02QBE 11415838 EC50 = 10400 nM T00890 C1SJY0 11470798 EC50 = 19000 nM T00890 C6VFI3 11492560 EC50 = 281.84 nM T00890 C85APY 11514348 EC50 = 57.54 nM T00890 CYFH61 11528793 EC50 = 199.53 nM T00890 CU8XZ6 11528819 EC50 = 151.36 nM T00890 C17BKW 11565047 EC50 = 309.03 nM T00890 CC43HE 11608532 EC50 = 9120.11 nM T00890 C8ECU6 11687485 EC50 = 1412.54 nM T00890 CI6Y4Q 11708383 EC50 = 257.04 nM T00890 CVFS35 11715531 EC50 = 100 nM T00890 CB8YL0 11739420 EC50 = 5100 nM T00890 CNC2Y3 11744994 EC50 = 398.11 nM T00890 CL7FM6 11817645 EC50 = 33000 nM T00890 C8CRY2 11961288 EC50 = 14.45 nM T00890 CDQ9F1 11992587 EC50 = 4466.84 nM T00890 CBH74R 11992588 EC50 = 6760.83 nM T00890 CXG82O 11992591 EC50 = 851.14 nM T00890 C3ITV5 11992592 EC50 = 8317.64 nM T00890 C1QP5H 11992688 EC50 = 5623.41 nM T00890 CAV6P2 11992689 EC50 > 10000 nM T00890 CP0T4C 11992788 EC50 > 10000 nM T00890 CSK39Y 11992789 EC50 > 10000 nM T00890 C0NC1J 11992790 EC50 = 8709.64 nM T00890 CU9J6V 13153555 EC50 = 18620.87 nM T00890 C5ZQ9X 15604637 EC50 = 140 nM T00890 CV3WB0 15604642 EC50 = 1300 nM T00890 CE7IR0 15605571 EC50 = 190 nM T00890 C7SOC8 16772244 EC50 < 10000 nM T00890 C6RPY7 16775596 EC50 = 6309.57 nM T00890 C4GN8A 17965902 EC50 = 1584.89 nM T00890 CS9IL0 22271415 EC50 = 7413.1 nM T00890 CDQK67 24955646 EC50 = 1120 nM T00890 CY32UX 28399894 EC50 = 41.69 nM T00890 CI4Z8C 28399946 EC50 = 51.29 nM T00890 CX9JP0 28400003 EC50 = 602.56 nM T00890 CB79PJ 28400019 EC50 = 933.25 nM T00890 COK4Y6 28400038 EC50 = 323.59 nM T00890 C7D6YH 28400046 EC50 = 1071.52 nM T00890 CR2F3V 28400056 EC50 = 269.15 nM T00890 C7HW2D 28400196 EC50 = 120.23 nM T00890 C5IG8A 28400380 EC50 = 100 nM T00890 C56JUZ 28400406 EC50 = 151.36 nM T00890 CSV67Z 43085192 EC50 = 363.08 nM T00890 CG92UM 43131474 EC50 = 1318.26 nM T00890 CFQ1W6 43187332 EC50 = 380.19 nM T00890 C9RA8K 43187344 EC50 = 3235.94 nM T00890 CJ91LE 43187366 EC50 = 602.56 nM T00890 C46TZC 43271417 EC50 = 52.48 nM T00890 CT1P7N 43271548 EC50 = 1621.81 nM T00890 CIV5T0 44433528 EC50 = 724.44 nM T00890 C4GC8E 44433529 EC50 = 3235.94 nM T00890 CJQP40 44433530 EC50 = 7585.78 nM T00890 CWJ8H0 44433532 EC50 = 12302.69 nM T00890 CFS0J5 44434363 EC50 = 3090.3 nM T00890 C3ISE8 44434380 EC50 = 72.44 nM T00890 C0FB2O 45268162 EC50 = 3981.07 nM T00890 CSQ82F 45269046 EC50 = 257.04 nM T00890 CDX01W 45269904 EC50 = 8912.51 nM T00890 CJC95S 45269912 EC50 = 141.25 nM T00890 C0R9FC 45271541 EC50 > 10000 nM T00890 C1HFL2 45272461 EC50 > 10000 nM T00890 CGW84J 51346919 EC50 = 300 nM T00890 CEDC82 59304608 EC50 = 67 nM T00890 CF70SZ 59343664 EC50 = 59 nM T00890 C2K3QR 135899171 IC50 = 33000 nM T00890 CC52JR 135899325 IC50 > 50000 nM T00890 C5MGD1 136127010 IC50 > 50000 nM T00890 D02GRY 11148966 EC50 = 4800 nM T00890 D0FF9F 6485181 EC50 = 11748.98 nM T00890 D0G8TM 11483496 EC50 = 370 nM T00890 D0IC7C 776421 EC50 = 41686.94 nM T00890 D0J7LY 11436345 EC50 = 180 nM T00890 D0K3LQ 11715556 EC50 = 29.51 nM T00890 D0T2KY 44250176 EC50 = 3.162 nM T00890 D0VE9G 2736690 EC50 = 398.11 nM T91180 D00HWO 19003 Ki = 500000 nM T91180 D01DSP 30699 Ki > 10000000 nM T91180 D01PLN 6024 Ki > 10000000 nM T91180 D02VFC 441199 Ki = 10000000 nM T91180 D04KTZ 6098 Ki = 2500000 nM T91180 D04QJD 135398742 IC50 = 431000 nM T91180 D04ZAH 43672 Ki > 30000000 nM T91180 D05JDR 5282242 Ki = 340000 nM T91180 D05UBX 42008 Ki = 28000000 nM T91180 D06KKS 38103 Ki = 9800000 nM T91180 D06OVY 5362065 Ki = 12000000 nM T91180 D06YHL 456255 Ki = 8100000 nM T91180 D07ACT 5479530 Ki > 30000000 nM T91180 D09CPR 6869 Ki = 21000000 nM T91180 D09KDN 33255 Ki > 30000000 nM T91180 D0A1CB 5479537 Ki > 30000000 nM T91180 D0D1HA 5742673 Ki > 30000000 nM T91180 D0MB8I 6196 Ki = 12000000 nM T91180 D0O5LU 47499 Ki = 12000000 nM T91180 D0PW7C 51039 Ki > 10000000 nM T91180 D0Q2AT 21319 Ki = 3200000 nM T91180 D0R2KJ 18381 Ki = 7200000 nM T91180 D0W6CA 6335986 Ki > 30000000 nM T91180 D0X9ZC 47965 Ki = 7200000 nM T91180 D0Y2IE 5479529 Ki = 26000000 nM T91180 D0Y7ZD 137 Ki = 790000 nM T91180 D0YA9Z 6249 Ki = 15000000 nM T91180 D0Z5EM 27447 Ki = 14000000 nM T91180 D00QAR 5904 Ki > 30000000 nM T91180 C0FD6Y 138 Ki = 17400000 nM T91180 CZ7DJ3 601 Ki = 120000 nM T91180 CW94UX 3238 Ki = 400000 nM T91180 C2M1AC 11161 EC50 = 580000 nM T91180 CXY67D 11163 EC50 = 480000 nM T91180 CHE36Y 70590 EC50 = 60000 nM T91180 CD6FT7 70910 Ki = 390000 nM T91180 CW59RX 76807 EC50 = 80000 nM T91180 C1W8YJ 78000 IC50 = 27400000 nM T91180 C7YC2T 80817 Ki = 110000 nM T91180 CZ0M7X 81721 Ki = 120000 nM T91180 C5F9KD 83525 Ki = 150000 nM T91180 C19KSO 85362 EC50 = 80000 nM T91180 CL13XP 87731 Ki = 25000000 nM T91180 C0V2WR 88184 IC50 = 80000 nM T91180 CTV32A 88656 IC50 = 250000 nM T91180 C7KR0D 92181 EC50 = 330000 nM T91180 CCOI47 92829 EC50 = 140000 nM T91180 CR71YD 92843 IC50 = 70000 nM T91180 C7E9ND 92946 EC50 = 60000 nM T91180 C57WLO 92953 EC50 = 130000 nM T91180 CS28ZP 96796 Ki = 4200000 nM T91180 CV98IP 96805 EC50 = 210000 nM T91180 C2TD8W 96814 IC50 = 70000 nM T91180 CPGC40 97050 Ki = 16000000 nM T91180 C3GQ5H 97054 EC50 = 260000 nM T91180 CQL18W 97363 Ki = 350000 nM T91180 C7LU0O 98153 Ki = 380000 nM T91180 CR01ON 99278 IC50 = 650000 nM T91180 C4BT8M 99719 EC50 = 230000 nM T91180 C4MKD1 101179 EC50 = 280000 nM T91180 CAP61W 101180 Ki = 480000 nM T91180 CIF3B6 107475 EC50 = 70000 nM T91180 CJ1W2Z 108985 Ki = 15000000 nM T91180 CBO69J 111104 Ki = 8300000 nM T91180 CJAG48 123715 Ki = 350000 nM T91180 CWQC87 128287 EC50 = 280000 nM T91180 CF08JC 128837 IC50 = 10900000 nM T91180 CDY34M 128841 Ki = 320000 nM T91180 C9RQF1 142765 EC50 = 270000 nM T91180 CH4KZ0 151004 Ki = 2500000 nM T91180 C7CN8P 151148 EC50 = 440000 nM T91180 C4FHS6 151956 IC50 = 7310000 nM T91180 C6QAR7 152264 Ki = 730000 nM T91180 CB9Q1L 168182 EC50 = 40000 nM T91180 C35FZA 194260 EC50 > 5000000 nM T91180 CYXW54 303942 Ki = 2900000 nM T91180 C47QLZ 439360 Ki = 2000000 nM T91180 C5ZW4M 439498 Ki = 200000 nM T91180 C0KG8H 439500 EC50 = 1000000 nM T91180 CE74WV 444109 EC50 = 250000 nM T91180 CW9JK0 471583 Ki = 410000 nM T91180 CZN6S9 743974 EC50 > 50118.72 nM T91180 C4HCS7 1549433 Ki = 140000 nM T91180 CUN54L 1549453 Ki = 90000 nM T91180 CQ6IO0 1551643 EC50 = 520000 nM T91180 C6HN0M 2282458 Ki = 20000 nM T91180 CZEY54 2965175 Ki = 16600000 nM T91180 CN52PM 3013625 EC50 = 130000 nM T91180 CA6E1H 3080576 EC50 = 750000 nM T91180 CT5W1J 3082062 Ki = 100000 nM T91180 C1SL9P 3152952 Ki = 12900000 nM T91180 CV02OY 3415972 Ki = 330000 nM T91180 C8TOU9 3496505 Ki = 14100000 nM T91180 C3N4DU 3811102 Ki = 340000 nM T91180 CWF6G0 4369021 Ki = 130000 nM T91180 C08JZU 4369395 IC50 = 660000 nM T91180 CQ5FT4 4670733 Ki = 2700000 nM T91180 CNRG81 5361871 Ki = 22000000 nM T91180 C4Z7MW 5460362 Ki > 30000000 nM T91180 CM47TY 5478845 Ki = 180000 nM T91180 CW75UJ 5479539 Ki > 30000000 nM T91180 CJHI21 5484352 EC50 = 80000 nM T91180 C2LQH6 5486959 Ki = 14000000 nM T91180 C6C1TR 5488196 Ki = 180 nM T91180 CZIC69 5488264 Ki > 30000000 nM T91180 CH5U2F 5491963 Ki = 320000 nM T91180 CF07VG 5496455 Ki = 90000 nM T91180 CTV2L1 6347578 Ki = 9500000 nM T91180 CM7DL9 6351946 Ki = 1900000 nM T91180 CV1E8W 6426709 IC50 > 16000000 nM T91180 C1Z7VT 6427003 Ki = 860000 nM T91180 CZ8LA0 6427006 IC50 = 8110000 nM T91180 C1A6GP 6427052 EC50 = 510000 nM T91180 COU6H0 6454191 Ki = 4900000 nM T91180 CG30YS 6713928 Ki = 13000000 nM T91180 C6KTO7 6992304 Ki = 200 nM T91180 CZT2G3 6992341 EC50 = 140000 nM T91180 C9W1MN 6992506 Ki = 250000 nM T91180 C1D9OY 6992569 Ki > 30000000 nM T91180 CIO6U0 6992638 Ki = 90000 nM T91180 C04HTR 6993090 Ki = 110000 nM T91180 CSK3A6 6993105 EC50 = 370000 nM T91180 CK3Q0Z 6993120 Ki = 50000 nM T91180 CGU7M1 6993122 Ki = 7000000 nM T91180 C0GH3W 6993389 Ki > 30000000 nM T91180 CY4FN2 6993401 EC50 = 100000 nM T91180 C7HIQ9 6998029 Ki = 140000 nM T91180 CMB48H 7009555 Ki = 100000 nM T91180 CVI1B7 7009579 Ki = 140000 nM T91180 C8EO3T 7009583 Ki = 5600000 nM T91180 CXH50C 7009600 Ki = 90000 nM T91180 C24NHU 7009616 IC50 = 310000 nM T91180 CW03QC 7009650 EC50 = 190000 nM T91180 CZ53RX 7009658 EC50 = 50000 nM T91180 C6T4PY 7010502 EC50 = 530000 nM T91180 C15XOM 7010504 Ki = 340000 nM T91180 C15TUA 7010588 EC50 = 100000 nM T91180 C8ZHS0 7015196 IC50 = 9110000 nM T91180 CQL26X 7015704 EC50 = 310000 nM T91180 CA2XY3 7016106 Ki = 210000 nM T91180 C49FKS 7016879 Ki = 6400000 nM T91180 CZNC34 7017967 Ki = 17000000 nM T91180 CB03SN 7019035 Ki = 70000 nM T91180 C0I2BU 7019105 IC50 = 130000 nM T91180 C0NV8K 7019964 Ki = 19000000 nM T91180 CIY21L 7020001 EC50 = 470000 nM T91180 CO1Y9H 7020029 EC50 = 420000 nM T91180 CLI20B 7020132 EC50 = 850000 nM T91180 C3C5HF 7020145 EC50 = 30000 nM T91180 C89NKE 7020215 EC50 = 210000 nM T91180 CJ67RM 7020642 Ki = 130000 nM T91180 CZ85ER 7021832 IC50 = 100000 nM T91180 CP4M1Q 7021854 EC50 = 240000 nM T91180 C36DHQ 7022320 EC50 = 320000 nM T91180 C2PR6I 7023107 EC50 = 400000 nM T91180 C5BER7 7023499 Ki = 14000000 nM T91180 CHY42A 7079450 IC50 = 9160000 nM T91180 C1XK6R 7408136 Ki = 1100000 nM T91180 C28NMU 7408195 Ki = 120000 nM T91180 C3QL4P 7408258 EC50 = 1600000 nM T91180 CZR45K 7408512 Ki = 150000 nM T91180 C70ZHW 7408741 Ki = 2000000 nM T91180 C7GYV3 9209431 IC50 > 16000000 nM T91180 CQT36A 9794235 Ki = 6300000 nM T91180 CNZA98 9795637 Ki = 160000 nM T91180 C69TPM 9815587 IC50 = 18200000 nM T91180 CVP24W 9818200 Ki = 100000 nM T91180 CDO9J0 9837272 Ki = 60000 nM T91180 C05KBM 9837455 Ki = 330000 nM T91180 CEI67G 9885148 Ki = 100000 nM T91180 CM3ZR9 9929972 Ki = 300000 nM T91180 CAS35Q 9949212 Ki = 280000 nM T91180 CQ54PR 10035657 Ki = 5400000 nM T91180 CV7Z4H 10159368 Ki = 240000 nM T91180 C42OVJ 10198309 IC50 = 1760000 nM T91180 CMA17B 10200042 Ki = 100000 nM T91180 CK6GJ8 10236791 Ki = 110000 nM T91180 CRY9H6 10403793 Ki = 19000 nM T91180 C9XZ8J 10668527 IC50 = 447000 nM T91180 CD0NB9 11179178 Ki = 68000 nM T91180 C75OSQ 11185657 Ki = 133000 nM T91180 C9P4QG 11218768 Ki = 140000 nM T91180 C3WV9X 11223118 Ki = 200000 nM T91180 CW8X3T 11233317 Ki = 905000 nM T91180 CS2NQ0 11279521 Ki = 100000 nM T91180 CL9RH2 11326774 Ki = 250000 nM T91180 C4SIT1 11334957 Ki = 417000 nM T91180 CD7OB3 11370352 Ki = 4300000 nM T91180 C10NFO 11380838 Ki = 90000 nM T91180 CVL2M9 11404267 Ki = 170000 nM T91180 CC3TH9 11622593 EC50 = 700000 nM T91180 C2ZGC0 11775677 Ki = 400 nM T91180 CTA35X 11807727 IC50 > 3000000 nM T91180 C1WG7A 11902901 Ki = 1600000 nM T91180 CVJG38 12546887 Ki = 3100000 nM T91180 CFOD02 13992965 Ki = 1500000 nM T91180 CT5L3G 14389323 Ki = 200000 nM T91180 COG9H6 14552273 EC50 = 190000 nM T91180 CL2IJ6 14602335 Ki = 4800000 nM T91180 CAF1H3 14855906 Ki = 1100000 nM T91180 C8DZ9I 15061422 IC50 = 7200000 nM T91180 CB5D0N 16122508 Ki > 30000000 nM T91180 CS0XZ6 18007123 Ki = 290000 nM T91180 CPMB46 20111857 Ki = 1200000 nM T91180 C3JOP4 20111874 Ki = 7000000 nM T91180 COY1R2 20111965 Ki = 250000 nM T91180 CGP4A0 20112232 Ki = 970000 nM T91180 CMLS62 21992231 IC50 > 3000000 nM T91180 CO0ZA3 24692381 Ki = 5620000 nM T91180 C5PD0B 24701102 Ki = 410000 nM T91180 CU89MI 24702462 Ki = 460000 nM T91180 CEQ05B 24704539 Ki = 7800000 nM T91180 C5YJT2 24905469 IC50 = 600000 nM T91180 CV7KI1 25260707 Ki = 90000 nM T91180 C05VZT 43579296 Ki = 890000 nM T91180 C01AQO 44266792 Ki = 39800 nM T91180 C5BAD6 44266833 Ki 26400 nM T91180 C5IKO4 44286974 IC50 = 2700000 nM T91180 CT7IE5 44368893 Ki = 11000000 nM T91180 C2EIU1 44369040 Ki = 2300000 nM T91180 CZ3IS8 44369126 Ki = 6900000 nM T91180 C20XAW 44398468 Ki = 90000 nM T91180 CMR2Y1 44398488 Ki = 140000 nM T91180 CR9VO6 44398504 Ki = 90000 nM T91180 C2BSJ7 44398506 Ki = 15000000 nM T91180 CFBU76 44398508 Ki = 1500000 nM T91180 CKF7U3 44398529 Ki = 5400000 nM T91180 CHZ0C9 44398536 Ki = 3100000 nM T91180 CX3SC4 44398561 Ki = 170000 nM T91180 C1EJR6 44398598 Ki = 330000 nM T91180 CJ4SM1 44398600 Ki = 110000 nM T91180 CQ28BM 44398612 Ki = 7900000 nM T91180 C43UBR 44398614 Ki = 1400000 nM T91180 CD7AV8 44398615 Ki > 30000000 nM T91180 C0RB4Q 44398622 Ki = 2900000 nM T91180 COT70A 44398636 Ki = 140000 nM T91180 CL13RT 44398643 Ki = 10000 nM T91180 CQ01IY 44412231 IC50 = 230000 nM T91180 CIX1B7 44818266 IC50 = 650000 nM T91180 CQMW07 44818267 IC50 = 630000 nM T91180 C31ZNT 44818268 IC50 = 2330000 nM T91180 CJ49RQ 45049835 Ki = 140000 nM T91180 C95ZVJ 46229343 IC50 = 390000 nM T91180 C3MK1D 46229344 IC50 = 630000 nM T91180 C9Q2YO 46832474 Ki = 210000 nM T91180 CB18ZD 46877033 IC50 = 96000 nM T91180 CDW5Y3 46877051 IC50 = 166000 nM T91180 CT7UQ8 46877054 IC50 = 142000 nM T91180 CO1FN8 46877101 IC50 = 477000 nM T91180 CT4H6I 46877108 IC50 = 537000 nM T91180 CAF4R0 46877141 IC50 = 300000 nM T91180 C4BP1Z 46877145 IC50 = 421000 nM T91180 CF2O9T 46877147 IC50 = 218000 nM T91180 CT0R6E 46877162 IC50 = 342000 nM T91180 C0PO2Q 46877167 IC50 = 282000 nM T91180 C8X4GA 46877180 IC50 = 260000 nM T91180 CV5LC8 53863424 Ki = 8300000 nM T91180 C95KAB 56670129 Ki = 257039578.3 nM T91180 CQ2M3R 56678253 IC50 = 121000 nM T91180 CR58UH 66262818 Ki = 60000 nM T91180 C97DOF 66724332 Ki = 160000 nM T91180 C9O1HB 70695689 Ki = 1400000 nM T91180 C93PDE 71396412 Ki = 1800000 nM T91180 C2AT7M 73345536 Ki = 120000 nM T91180 C7EVI9 73345537 Ki = 130000 nM T91180 C2P3HE 73345599 Ki = 20000 nM T91180 CL2XH0 73354636 Ki = 20000 nM T91180 CCH96U 73354637 Ki = 160000 nM T91180 C1AU9W 145948213 Ki = 245470891.6 nM T91180 C4OAT5 145948219 Ki = 323593656.9 nM T91180 CVP8X5 145948220 Ki = 251188643.2 nM T91180 CF30AZ 145948221 Ki = 46773514.13 nM T91180 C10EQW 145948223 Ki = 123026877.1 nM T91180 C1TLF5 155550193 IC50 = 2900000 nM T91180 CWU63B 137672 Ki = 7300000 nM T91180 CX8JW1 141894 Ki = 4800000 nM T91180 C9UJF7 18400028 Ki = 310000 nM T91180 CM5XD8 21428097 Ki = 10000 nM T91180 C1V4EN 21708023 Ki = 9100000 nM T91180 CR89ZX 263465 Ki > 30000000 nM T91180 C8DX3P 44369036 Ki = 2800000 nM T91180 C3BK2G 44369181 Ki = 330000 nM T91180 CC62RB 7020236 Ki = 32000000 nM T91180 CV2P6M 9899097 Ki = 1200000 nM T91180 D0Q3VU 93131 EC50 = 540000 nM T91180 D0XR4J 85169 EC50 = 30000 nM T65561 C6HA8E 5388709 IC50 > 30000 nM T65561 C8W2QA 6439099 IC50 = 3700 nM T65561 CQSZ72 90675942 IC50 = 14000 nM T65561 CTBD74 90675943 IC50 = 7900 nM T65561 CM12LR 102597975 IC50 = 1600 nM T65561 CW9P6A 145964460 IC50 = 29000 nM T65561 CQR49Z 145965116 IC50 = 11000 nM T65561 CR6L2G 145967358 IC50 = 24000 nM T65561 CHXE25 145978207 IC50 = 17000 nM T65561 D08BMM 6312649 IC50 = 4900 nM T65561 D0R9CF 11302540 IC50 = 130 nM T57253 CNMB45 122185 EC50 > 100000 nM T57253 CO1NZ5 11539085 IC50 = 800 nM T57253 CIA94D 16158367 EC50 = 50 nM T57253 C84ZJU 25208742 EC50 = 26302.68 nM T57253 C5YXN8 25208743 EC50 = 19952.62 nM T57253 C9HU3K 25208744 EC50 = 2691.53 nM T57253 CR8YK2 25208745 EC50 = 8128.31 nM T57253 C69EKG 25208894 EC50 = 131.83 nM T57253 CZB37J 25208895 EC50 = 398.11 nM T57253 C9RT2Y 25208898 EC50 = 123.03 nM T57253 CI95DJ 25209047 EC50 = 295.12 nM T57253 C6M2BT 25209048 EC50 = 2137.96 nM T57253 CN06PX 25209050 EC50 = 19.95 nM T57253 CKPY96 25209191 EC50 = 20892.96 nM T57253 CJTU64 25209192 EC50 = 10964.78 nM T57253 CA8SQ7 25209193 EC50 = 588.84 nM T57253 C8U0MT 25209194 EC50 = 144.54 nM T57253 C4XQ3N 25209354 EC50 = 4168.69 nM T57253 CKS65O 25209355 EC50 = 288.4 nM T57253 CR1K8B 25209356 EC50 = 23.99 nM T57253 CLKT16 25209357 EC50 = 52.48 nM T57253 C1X2EP 25209534 EC50 = 81.28 nM T57253 C8UY1L 25209535 EC50 = 107.15 nM T57253 CJ9F2A 25209536 EC50 = 5754.4 nM T57253 C5VO1W 25209537 EC50 = 7079.46 nM T57253 C2RTJ1 25209704 EC50 = 32359.37 nM T57253 CDF83Q 25209705 EC50 = 6.31 nM T57253 C5NS6H 44581972 EC50 = 8317.64 nM T57253 CK8Z1P 44581973 EC50 = 4073.8 nM T57253 C3UQ9Z 44581974 EC50 = 125.89 nM T57253 C6KLM2 54580023 IC50 = 8060 nM T57253 C9B7HW 54580024 IC50 = 40 nM T57253 CN83VE 54580025 IC50 = 88 nM T57253 C7T9IX 54580026 IC50 = 14 nM T57253 CV7NF5 54581018 IC50 = 24 nM T57253 CGWM27 54581019 IC50 = 295 nM T57253 CQ56JN 54581020 IC50 = 108 nM T57253 CVD14I 54584003 IC50 = 640 nM T57253 CUQR37 54584004 IC50 = 301 nM T57253 C7BD8E 54584942 IC50 = 758 nM T57253 C6O8XI 54584943 IC50 = 20 nM T57253 CMKH64 54584944 IC50 = 22 nM T57253 CSJ7Z8 54584945 IC50 = 244 nM T57253 C1IS8L 54585912 IC50 = 530 nM T57253 C09ACT 54585913 IC50 = 330 nM T57253 COI6N1 54586326 IC50 = 77 nM T57253 C4J8EG 118717463 EC50 > 100000 nM T57253 C6TBR9 118717464 EC50 > 100000 nM T57253 C8Z5CS 118717465 EC50 > 100000 nM T57253 C85ECX 118717466 EC50 > 100000 nM T57253 CI0W7X 118717467 EC50 > 100000 nM T57253 C0BH8P 118717468 EC50 > 100000 nM T57253 CL9ZY7 139030531 EC50 = 50 nM T57253 CXRH34 155511165 EC50 = 5200 nM T57253 CQI28S 155517690 EC50 = 290 nM T57253 C9V4QT 155518019 EC50 = 920 nM T57253 C9CU8K 155518320 EC50 > 100000 nM T57253 CEN9G8 155523607 EC50 = 300 nM T57253 CF5BP3 155524924 EC50 = 150 nM T57253 CIQD10 155530228 EC50 = 1900 nM T57253 CG7D3Q 155530554 EC50 = 3300 nM T57253 CE31WQ 155536163 EC50 = 3700 nM T57253 CAP07B 155541652 EC50 = 5200 nM T57253 CD9U4P 155542939 EC50 = 680 nM T57253 C4WIF6 155543843 EC50 = 100 nM T57253 CDE89A 155544956 EC50 = 3600 nM T57253 CY6RU0 155546489 EC50 = 23000 nM T57253 CQ2XN8 155551191 EC50 = 160 nM T57253 CJ31MZ 155563230 EC50 = 2100 nM T57253 C8XSU5 155566258 EC50 = 2200 nM T57253 CIH8N4 155567014 EC50 > 100000 nM T57253 CB1IO9 135407930 EC50 = 63.1 nM T57253 C6IYM1 135407979 EC50 = 630.96 nM T57253 C34ABJ 136036237 EC50 = 316.23 nM T57253 CLUV03 136036258 EC50 = 2511.89 nM T57253 C9YAL3 136036260 EC50 = 1258.93 nM T57253 C8Y7FX 136036261 EC50 = 199.53 nM T57253 C3H7NG 136036262 EC50 = 316.23 nM T57253 D02XPB 23646462 EC50 = 510 nM T57253 D08UWO 53320361 EC50 > 100000 nM T89323 D03QLG 9917013 IC50 = 2 nM T89323 D0E3TC 44259 IC50 = 2.69 nM T89323 C18WEB 490561 IC50 = 45 nM T89323 CK21EQ 9796713 IC50 = 364 nM T89323 CJH69P 9840393 IC50 = 2088 nM T89323 CR3DA5 9939328 IC50 = 89 nM T89323 CHB35P 10604501 IC50 = 627 nM T89323 CJ4BN2 10626594 IC50 = 16 nM T89323 CGP93J 10745853 IC50 = 20 nM T89323 C4NO7Y 11809063 IC50 = 2664 nM T89323 C20DST 16105503 IC50 = 3447 nM T89323 CCN62F 16105510 IC50 = 339 nM T89323 C3E7RP 44284203 IC50 = 28 nM T89323 C8FY7N 44284204 IC50 = 140 nM T89323 COH62U 60097413 IC50 > 10000 nM T89323 C1MR8Q 60097495 IC50 > 10000 nM T89323 CV63UL 67240318 IC50 > 10000 nM T89323 CZ4BX1 72547959 IC50 = 767 nM T89323 CQ2OB9 90292687 IC50 = 5150 nM T89323 CHI39S 90292823 IC50 = 7880 nM T89323 CJQ5N6 91936970 IC50 > 10000 nM T89323 CXC69T 137321158 IC50 = 50 nM T89323 CI1E8V 137634241 IC50 = 4550 nM T89323 C6VB3O 145925651 IC50 >= 5000 nM T89323 CV9QD6 145968243 IC50 = 46 nM T89323 C2MD1Q 155513187 IC50 > 10000 nM T89323 C86HPW 155518524 IC50 = 18000 nM T89323 D07ADX 54764565 IC50 = 42 nM T89323 D07IHM 9823787 IC50 = 1855 nM T89323 D09QBA 23378546 IC50 = 1582 nM T89323 D0J3LR 11634725 Ki > 10000 nM T89323 D0N4LR 53469448 IC50 = 452 nM T73189 C8M6NW 44329079 IC50 = 200 nM T73189 C6WOM8 44329152 IC50 = 70 nM T73189 CIT4Z0 44329153 IC50 = 100 nM T73189 CW57TV 44329424 IC50 = 3000 nM T73189 CMZ32C 44329425 IC50 = 80 nM T73189 C14JVE 44329430 IC50 = 260 nM T73189 C1DKT9 44329431 IC50 = 70 nM T73189 C09UJF 44329432 IC50 = 35 nM T73189 CU6TF7 44329459 IC50 = 4000 nM T73189 C69LNC 44329497 IC50 = 600 nM T73189 CU5HX0 44329498 IC50 = 150 nM T73189 CF78XJ 44329510 IC50 = 90 nM T73189 CE3W7H 44329537 IC50 = 800 nM T73189 C21OLE 44329538 IC50 = 50 nM T73189 C6UK9W 44329659 IC50 = 200 nM T73189 CXIR40 44329660 IC50 = 40 nM T73189 C9QV0N 44329674 IC50 = 2900 nM T73189 C6CJ7B 44329680 IC50 = 30 nM T73189 CC4XB1 44329681 IC50 = 100 nM T73189 C8OF7U 44329682 IC50 > 5000 nM T73189 CV4ZJ0 44329743 IC50 = 450 nM T73189 CT5RC4 44329744 IC50 = 550 nM T73189 CM98VF 44329745 IC50 = 60 nM T73189 CPM1A0 44329776 IC50 > 10000 nM T73189 CEYF26 44329777 IC50 = 100 nM T73189 C9RIV3 44329778 IC50 = 70 nM T73189 C5WB4A 44329785 IC50 = 200 nM T73189 C0GRU3 44329786 IC50 = 120 nM T73189 C7OJ0Q 44329787 IC50 = 150 nM T02653 D04DJN 10635 IC50 = 360 nM T02653 D07BSQ 5994 IC50 = 14 nM T02653 D0D1SG 5755 EC50 = 0.002 nM T02653 D0EP0C 5833 IC50 = 1.6 nM T02653 D0G8BV 6450278 Ki = 37 nM T02653 D0I1LH 5839 EC50 = 0.18 nM T02653 D0IT2G 5743 Ki = 0.36 nM T02653 D0Q4SD 443872 IC50 = 63.1 nM T02653 D0Y7IU 5281004 EC50 = 4.8 nM T02653 D0Y7JU 9854489 IC50 = 166 nM T02653 D0Z4EI 55245 IC50 = 590 nM T02653 D00JFE 56941241 IC50 > 1000 nM T02653 D01SYU 10026128 IC50 = 10000 nM T02653 D05RZE 42636651 Ki = 0.33 nM T02653 D07MON 5311505 IC50 = 470 nM T02653 D0SZ1G 121248172 IC50 > 38000 nM T02653 D0X9YP 67041274 IC50 > 10000 nM T02653 D0TH6M 25204767 EC50 > 10000 nM T02653 D0W1XE 91827457 IC50 > 10000 nM T02653 D02KAU 46871935 IC50 = 9 nM T02653 D03KTE 16750192 Ki > 10000 nM T02653 D09UFV 24825740 IC50 > 5000 nM T02653 D0W5RL 9577221 IC50 = 1600 nM T02653 C59UQE 6279 IC50 = 1197 nM T02653 C2O8KM 101788 EC50 = 50 nM T02653 C40YBS 444036 IC50 = 149 nM T02653 C8AMD7 2848661 IC50 = 460 nM T02653 CLBV35 3699263 IC50 = 850 nM T02653 C43BVE 3816305 IC50 = 1070 nM T02653 CDCK27 5185174 IC50 = 1400 nM T02653 C16ZSG 6439929 Ki = 39 nM T02653 C7REX1 9805004 IC50 = 38 nM T02653 CV87EA 9820084 IC50 = 290 nM T02653 C8A3WG 9820510 Ki > 10000 nM T02653 C06RXB 9821393 Ki = 1682 nM T02653 CD9S5P 9825465 Ki = 3838 nM T02653 CE62WD 9839013 IC50 > 1000 nM T02653 CBS8M2 9839134 IC50 = 2369 nM T02653 C92CPK 9841404 Ki > 10000 nM T02653 CK7UC3 9841413 Ki > 10000 nM T02653 C7P6XH 9842832 Ki > 10000 nM T02653 C7RS9U 9846657 Ki > 5000 nM T02653 CERF28 9861044 Ki > 10000 nM T02653 C3K4EU 9862027 Ki > 10000 nM T02653 CEM27C 9885473 IC50 = 3000 nM T02653 C6B9CZ 9888873 IC50 = 160 nM T02653 CZ5R9B 9890023 Ki = 493 nM T02653 CJ7U3R 9904286 IC50 > 10000 nM T02653 C6SWK1 9904610 IC50 = 2492 nM T02653 CTI1J8 9905296 Ki > 10000 nM T02653 CE1TK2 9908041 IC50 > 10000 nM T02653 CMJG42 9921530 IC50 > 10000 nM T02653 C39EXP 9933936 IC50 = 454 nM T02653 C24FUO 9943699 IC50 = 1386 nM T02653 CCSX75 9949772 IC50 = 1500 nM T02653 CKU64T 9952569 IC50 = 333 nM T02653 CW0ED9 9953456 IC50 = 681 nM T02653 C95CAN 9978625 Ki = 0.967 nM T02653 C1QP8T 9993897 IC50 = 2000 nM T02653 C4V6RF 9998996 IC50 > 5000 nM T02653 CC4WY6 10024990 IC50 = 1000 nM T02653 CSM0W3 10026120 IC50 > 2000 nM T02653 CFY67M 10070808 IC50 = 2219 nM T02653 C9T4HR 10071810 IC50 = 1100 nM T02653 CQ3LD1 10091351 IC50 = 1600 nM T02653 C16HAK 10094808 IC50 > 2000 nM T02653 CR0DX5 10126475 IC50 > 1130 nM T02653 CHS18G 10126476 IC50 > 2000 nM T02653 CR0BP6 10126871 IC50 = 380 nM T02653 CV5PQ0 10126940 IC50 = 500 nM T02653 CVF40M 10127159 IC50 = 350 nM T02653 C3CRZ1 10127269 IC50 = 450 nM T02653 CPB60D 10127340 IC50 = 760 nM T02653 CKMW98 10128037 IC50 = 585 nM T02653 C1GI3D 10150743 IC50 = 220 nM T02653 CZKF71 10150825 IC50 = 400 nM T02653 CYR0U5 10150851 IC50 > 2000 nM T02653 CVO1F7 10151165 IC50 = 405 nM T02653 C6EC1P 10151186 IC50 = 405 nM T02653 CQ14RM 10151357 IC50 = 535 nM T02653 CW4Y2K 10151995 IC50 = 1650 nM T02653 C0MX7K 10157532 IC50 = 893 nM T02653 CL0U4N 10172897 IC50 = 400 nM T02653 CG0VH8 10173354 IC50 = 1250 nM T02653 CU6D8W 10173525 IC50 = 170 nM T02653 C8L7HJ 10179031 IC50 = 683 nM T02653 C41YRZ 10194268 IC50 > 740 nM T02653 CX4F7Z 10194607 IC50 > 2000 nM T02653 CV0LE4 10194889 IC50 > 1000 nM T02653 C3O7WH 10215978 IC50 = 1350 nM T02653 C1SG4N 10216152 IC50 > 1420 nM T02653 CD0YT7 10216465 IC50 = 940 nM T02653 C1FGX9 10216535 IC50 = 415 nM T02653 CW7QX2 10216536 IC50 = 720 nM T02653 CG9OH4 10216697 IC50 = 1050 nM T02653 CXN4W1 10216788 IC50 = 1100 nM T02653 CUGN98 10217411 IC50 = 910 nM T02653 CJ9BE0 10222329 IC50 = 651 nM T02653 C84SRT 10223610 IC50 = 2154 nM T02653 CUYO17 10237223 IC50 > 1300 nM T02653 CWYK62 10238100 IC50 = 435 nM T02653 C1R8GY 10238297 IC50 = 900 nM T02653 CNB1V3 10238624 IC50 = 190 nM T02653 CPGF94 10238831 IC50 > 2000 nM T02653 C2AZH1 10238961 IC50 = 175 nM T02653 CSA4R3 10252455 IC50 > 2000 nM T02653 C7EGH2 10252527 IC50 = 120 nM T02653 CR59SC 10271193 IC50 = 22897 nM T02653 CPIS57 10271557 IC50 = 2252 nM T02653 CUQC81 10287415 IC50 > 1000 nM T02653 C5RC7X 10287444 IC50 = 510 nM T02653 CJT2G8 10287863 IC50 = 1400 nM T02653 C1M6WY 10288006 IC50 = 320 nM T02653 CO6UP3 10288155 IC50 = 875 nM T02653 C6C2IK 10288565 IC50 = 195 nM T02653 CNEO49 10289020 IC50 = 104 nM T02653 CLJU03 10298892 Ki = 3914 nM T02653 C9UYG8 10309447 IC50 > 1050 nM T02653 C8FM2D 10309755 IC50 = 1800 nM T02653 C1OV7M 10309756 IC50 = 715 nM T02653 C9TI4A 10310063 IC50 = 1035 nM T02653 CP9AE0 10310476 IC50 > 512 nM T02653 CV52EN 10310809 IC50 = 140 nM T02653 CR1L5N 10311251 IC50 = 104 nM T02653 CX7WS4 10316069 IC50 = 354 nM T02653 CQP1Y7 10340204 IC50 = 1525 nM T02653 CEJ78I 10365592 IC50 > 2000 nM T02653 CDBZ06 10372181 IC50 = 120 nM T02653 C14AIB 10384345 IC50 = 970 nM T02653 CZ5CJ3 10423330 IC50 > 10000 nM T02653 C5I3BG 10428464 Ki = 12 nM T02653 C1KE6C 10446402 IC50 = 2050 nM T02653 C0NT9D 10454007 IC50 > 5000 nM T02653 C85RBN 10474264 IC50 > 2000 nM T02653 CUL8O4 10475384 IC50 > 5000 nM T02653 CPX65M 10477088 IC50 = 130 nM T02653 C5AP6C 10503520 IC50 > 10000 nM T02653 CBEC38 10596252 IC50 = 1000 nM T02653 CC8T7J 10598305 IC50 = 1062 nM T02653 CO3V0S 10622594 IC50 = 977 nM T02653 C02ZMG 10643956 IC50 = 748 nM T02653 CYNG45 10668755 IC50 > 10000 nM T02653 CYRQ10 10691647 Ki = 1100 nM T02653 CVD2Y9 10717098 IC50 > 10000 nM T02653 CAT1X8 10741366 IC50 = 1068 nM T02653 CB3JD0 10763832 IC50 = 1358 nM T02653 C07BOR 10787258 IC50 = 2035 nM T02653 C1CRQ5 10811045 IC50 > 10000 nM T02653 CN1H5Z 10832792 IC50 = 1592 nM T02653 CHU9A4 10873317 IC50 = 334 nM T02653 CHU10G 10960295 IC50 = 1850 nM T02653 C6LYG7 11090322 IC50 > 1000 nM T02653 CXS6J7 11155441 Ki = 10 nM T02653 CQUV78 11176984 IC50 = 23 nM T02653 CL97OU 11212803 IC50 = 540 nM T02653 C4U0DF 11213029 Ki = 980 nM T02653 CRN4V2 11232136 IC50 > 3000 nM T02653 C8XPZ4 11269445 IC50 > 2000 nM T02653 C4HNB8 11269886 IC50 = 1050 nM T02653 CC0XI4 11279959 IC50 = 440 nM T02653 C4SC0W 11281576 IC50 > 5000 nM T02653 C8YL6K 11282486 IC50 = 1700 nM T02653 CUX0S2 11282904 Ki = 21 nM T02653 CIY9H5 11291999 IC50 = 1800 nM T02653 C0IQ9K 11304445 IC50 = 160 nM T02653 C0XUF2 11305564 IC50 > 5000 nM T02653 CXC9G3 11327341 IC50 > 2000 nM T02653 CT9Y4O 11339440 IC50 = 2300 nM T02653 C8FQ9B 11375180 IC50 = 21000 nM T02653 CP2DL0 11377050 IC50 = 1000 nM T02653 C76VYN 11382721 IC50 > 2000 nM T02653 CV4RO2 11384310 IC50 = 48 nM T02653 CXW40M 11384346 IC50 > 2000 nM T02653 CU7IE0 11410199 IC50 = 690 nM T02653 CO20QH 11416730 IC50 = 155 nM T02653 C5WO0U 11429662 IC50 > 5000 nM T02653 CD2Q3F 11474917 IC50 = 83 nM T02653 CC75NQ 11477616 Ki = 430 nM T02653 CQ62KS 11485693 IC50 > 3000 nM T02653 C9Q1NY 11494167 Ki = 32 nM T02653 CFLQ08 11495227 IC50 = 320 nM T02653 C03NYX 11495549 IC50 = 90 nM T02653 CR40IH 11516847 IC50 = 1800 nM T02653 CP4F8X 11517412 IC50 = 280 nM T02653 C2PB6Z 11530605 Ki = 930 nM T02653 C1R6DC 11531942 IC50 = 140 nM T02653 CZ1HA3 11538472 IC50 = 615 nM T02653 CFC1Z4 11538799 IC50 = 1100 nM T02653 CBK60G 11559947 IC50 > 2000 nM T02653 C1D9YS 11560003 IC50 > 2000 nM T02653 CB37YF 11566981 Ki = 145 nM T02653 C8WJ2F 11567609 IC50 = 780 nM T02653 C0SCT6 11588584 IC50 = 810 nM T02653 C3MW1D 11589982 IC50 = 220 nM T02653 C03QYZ 11590471 IC50 = 110 nM T02653 CAO2P1 11596392 IC50 > 2000 nM T02653 CSB97O 11617028 Ki = 21 nM T02653 CRL3A7 11632925 IC50 = 120 nM T02653 CQB0E3 11633482 IC50 = 65 nM T02653 C9DNG1 11640164 IC50 = 580 nM T02653 C1RJ3I 11646689 IC50 = 1000 nM T02653 CX3L5S 11647533 IC50 = 80 nM T02653 C4S5RG 11655053 IC50 = 175 nM T02653 CDOZ32 11661172 IC50 = 590 nM T02653 C0LEZ3 11667800 Ki = 890 nM T02653 C5XEN0 11668719 IC50 = 220 nM T02653 CZPK72 11682989 IC50 = 80 nM T02653 CCK83U 11690269 IC50 = 160 nM T02653 CY07JH 11696378 IC50 > 2000 nM T02653 CBU02W 11696959 IC50 = 640 nM T02653 C2S9IT 11697271 IC50 = 1900 nM T02653 CGR32I 11697882 IC50 = 340 nM T02653 C75IBX 11704529 IC50 = 90 nM T02653 CGX54N 11704756 IC50 = 210 nM T02653 CO2N1W 11710364 IC50 = 1550 nM T02653 CZ52YQ 11710766 IC50 < 500 nM T02653 C8OPA1 11710962 IC50 = 855 nM T02653 CW3N8H 11711766 IC50 = 280 nM T02653 COEU05 11719039 IC50 = 100 nM T02653 CZ0B7H 11731863 IC50 = 1900 nM T02653 CQO76Z 11741168 IC50 > 2000 nM T02653 C87YNC 11741891 IC50 = 150 nM T02653 CH92VI 11743259 IC50 = 310 nM T02653 C5HLU8 11750204 IC50 = 380 nM T02653 CY1F4I 11752649 Ki = 670 nM T02653 CQU0E7 11774868 IC50 = 435 nM T02653 C4U8KY 12085089 IC50 = 162 nM T02653 C14LTD 15463551 IC50 > 1000 nM T02653 C3QOV0 16099227 IC50 = 430 nM T02653 CW6LO1 16099229 IC50 > 2000 nM T02653 C2R4PK 16099231 IC50 = 450 nM T02653 C9KM7X 16099232 IC50 = 1900 nM T02653 C05CYN 16099234 IC50 = 1600 nM T02653 CJQ8A1 16099236 IC50 = 450 nM T02653 CA72YW 16099237 IC50 > 2000 nM T02653 CS07DB 16099238 IC50 = 98 nM T02653 C42ESN 16099240 IC50 = 580 nM T02653 CMZ91J 16099242 IC50 > 2000 nM T02653 CF69RC 16099243 IC50 > 2000 nM T02653 C60GEM 16099245 IC50 = 1500 nM T02653 CE48CS 16099246 IC50 = 620 nM T02653 CTF2M7 16099247 IC50 = 130 nM T02653 CX9BK2 16099248 IC50 = 775 nM T02653 CN6PA9 16099249 IC50 = 350 nM T02653 C9Z6AK 16099250 IC50 = 120 nM T02653 C5Z8HR 16099251 IC50 = 91 nM T02653 CWK76M 16099252 IC50 = 880 nM T02653 C3BU9M 16216822 IC50 = 290 nM T02653 C1Q5SV 16220168 IC50 = 510 nM T02653 CH6CN0 16658901 Ki > 10000 nM T02653 CU9LS2 16661702 EC50 = 5000 nM T02653 C1UY8J 16666386 IC50 > 1000 nM T02653 CWK35C 16730429 IC50 = 8700 nM T02653 CSKX58 17758233 Ki = 410 nM T02653 C7CPW9 17758234 Ki = 48 nM T02653 CI5KT6 17758236 Ki = 42 nM T02653 C3FP7L 17921933 IC50 = 3162 nM T02653 CX03YG 18188955 IC50 = 1220 nM T02653 CR19ST 18512166 IC50 = 310 nM T02653 CEN14G 18512334 IC50 = 4000 nM T02653 CS9CI5 18551230 IC50 = 30 nM T02653 CBI64N 18551237 IC50 = 130 nM T02653 C5ZYJ0 20231824 Ki = 952 nM T02653 CEH7V5 20786216 IC50 > 1000 nM T02653 C97WCO 21941658 IC50 = 1.259 nM T02653 CCI89R 21948853 IC50 > 1000 nM T02653 CB2SF4 21948904 IC50 > 1000 nM T02653 C2ZP7V 22218142 IC50 = 1500 nM T02653 C1QTK4 22398492 IC50 = 240 nM T02653 C6CSB4 22398502 IC50 > 2000 nM T02653 CR8N1E 22398506 IC50 = 1420 nM T02653 CM83TU 22398533 IC50 = 265 nM T02653 C34LHW 22398559 IC50 = 910 nM T02653 CJBW90 22398592 IC50 > 2000 nM T02653 CEJ65O 22398627 IC50 = 415 nM T02653 CZI4C6 24739672 Ki = 1000 nM T02653 CS23KY 24739834 Ki = 1390 nM T02653 C1M9QG 24739836 Ki = 1770 nM T02653 CG5SJ0 24739997 Ki = 1490 nM T02653 C7Z1HW 24740156 Ki = 1440 nM T02653 CTE1N2 24748569 EC50 > 10000 nM T02653 C4WYE7 24749678 Ki = 1.56 nM T02653 CY2JS4 24749684 Ki = 1.51 nM T02653 C2QHO3 24749808 Ki = 0.319 nM T02653 C5S6JN 24780149 IC50 > 1000 nM T02653 CW5TJ7 24781731 IC50 > 1000 nM T02653 C1JTW2 24851053 Ki = 0.342 nM T02653 CC53XL 24860583 Ki > 3000 nM T02653 C58RHY 24883011 IC50 = 80 nM T02653 CW35CK 24883012 IC50 = 41 nM T02653 C3SC0V 24883054 IC50 = 76 nM T02653 C4SA6C 24883055 IC50 = 15 nM T02653 C5LZK2 24895096 IC50 = 1350 nM T02653 COGP96 24936313 IC50 > 5000 nM T02653 CVY09S 24936449 IC50 > 5000 nM T02653 C06PDG 24952192 EC50 > 5000 nM T02653 CG1CF9 24952193 EC50 > 5000 nM T02653 CZC7L8 24953162 IC50 > 10000 nM T02653 C4W7BN 24954947 IC50 > 10000 nM T02653 C6XC2R 24954951 IC50 > 20000 nM T02653 CYES17 24957737 Ki > 3000 nM T02653 C83YKB 24961057 Ki > 1000 nM T02653 CIGM27 24983460 IC50 = 280 nM T02653 CHY0D7 25013322 IC50 > 10000 nM T02653 C0TPS5 25013653 IC50 > 10000 nM T02653 CWU91M 25013811 IC50 > 10000 nM T02653 CSH29L 25013812 IC50 > 10000 nM T02653 C7QCX0 25052023 IC50 = 2.4 nM T02653 CAW8M0 25070694 IC50 = 2800 nM T02653 C21XDY 25145083 Ki > 10000 nM T02653 CS6JQ1 25167502 Ki = 155 nM T02653 C0XPW9 25168896 IC50 = 340 nM T02653 CUL27D 25168900 IC50 = 260 nM T02653 CEV2D7 25205475 IC50 = 260 nM T02653 C9S0ZW 25205477 IC50 = 330 nM T02653 C49KHR 25206116 IC50 = 510 nM T02653 C9FM2U 42642501 Ki <= 10 nM T02653 CXZ35T 44193145 Ki = 656 nM T02653 C2MOF7 44193146 Ki = 378 nM T02653 CWR6X1 44193147 Ki = 2250 nM T02653 C3JOW4 44193245 Ki = 1470 nM T02653 CHGI03 44251606 IC50 = 475 nM T02653 C0OA6M 44264483 IC50 > 10000 nM T02653 COCE32 44264569 IC50 > 10000 nM T02653 CI0TN2 44264577 IC50 > 10000 nM T02653 CXOR54 44264579 IC50 > 10000 nM T02653 C01HSQ 44264588 IC50 > 10000 nM T02653 CDB54J 44305270 IC50 > 1000 nM T02653 C0XLN6 44305556 IC50 > 1000 nM T02653 C1UK4M 44305720 IC50 = 1889 nM T02653 CH4PU5 44305819 IC50 = 2484 nM T02653 C6N1AR 44305929 IC50 2871 nM T02653 C73CXK 44354006 IC50 = 363 nM T02653 C0N3TD 44354884 IC50 = 2700 nM T02653 CPQ2A6 44354885 IC50 = 1000 nM T02653 CM0G1V 44354886 IC50 = 2000 nM T02653 CL6G3Q 44355066 IC50 = 2100 nM T02653 CSAU31 44377064 IC50 > 10000 nM T02653 C7H9NC 44377081 IC50 > 10000 nM T02653 C60DYH 44377090 IC50 = 2000 nM T02653 CVH2R3 44377098 IC50 = 2900 nM T02653 CYLI63 44377110 IC50 > 10000 nM T02653 CQX39I 44377356 IC50 = 570 nM T02653 C9FJW4 44377382 IC50 = 1900 nM T02653 C13SYV 44396250 Ki = 300 nM T02653 CB1P0S 44396251 Ki = 80 nM T02653 CHY1C3 44396271 Ki = 590 nM T02653 C29MBI 44396272 Ki = 310 nM T02653 C4TQ6N 44396282 Ki = 440 nM T02653 CH2Y3L 44396283 Ki = 190 nM T02653 CWZB52 44396284 Ki = 850 nM T02653 CD80LM 44396296 Ki > 1000 nM T02653 C6SI5L 44396297 Ki > 1000 nM T02653 CR4H1E 44396316 Ki = 510 nM T02653 C45LRH 44396317 Ki = 140 nM T02653 C5JG6H 44396330 Ki > 1000 nM T02653 CA8V4G 44396331 Ki > 1000 nM T02653 C57CPQ 44396332 Ki = 310 nM T02653 CXHF58 44403036 IC50 = 215 nM T02653 C6JNI4 44403038 IC50 = 60 nM T02653 C45SOW 44403039 IC50 = 315 nM T02653 CXZ4S3 44426781 Ki = 3490 nM T02653 C8HO4K 44426782 Ki = 585 nM T02653 C0FEN3 44426790 Ki = 298 nM T02653 C19MJP 44426793 Ki = 527 nM T02653 C1ZDA4 44426795 Ki = 1270 nM T02653 CIOW01 44431179 IC50 = 520 nM T02653 C3SJ5V 44433504 Ki = 7.5 nM T02653 C2SCP7 44435606 IC50 = 1600 nM T02653 CH5E3L 44435611 IC50 > 1300 nM T02653 CDO62N 44435656 IC50 = 650 nM T02653 C9TP4C 44435662 IC50 = 345 nM T02653 C19TMW 44435663 IC50 = 730 nM T02653 C90WUC 44435667 IC50 = 430 nM T02653 CHFB89 44435668 IC50 = 300 nM T02653 C8IWK2 44435669 IC50 = 250 nM T02653 CYG7X4 44473146 IC50 > 10000 nM T02653 CR5SI0 44476535 EC50 > 10000 nM T02653 CM29JD 44516036 IC50 > 10000 nM T02653 CR19IH 44543858 IC50 > 2000 nM T02653 C05HEP 44543860 IC50 > 2000 nM T02653 C45ZHO 44543969 IC50 > 2000 nM T02653 C25OXZ 44544094 IC50 > 2000 nM T02653 C7JIF6 44544321 IC50 > 2000 nM T02653 CF6V4G 44563171 EC50 > 10000 nM T02653 C8BGL6 44585565 IC50 > 3000 nM T02653 CIJP09 44605898 IC50 > 10000000 nM T02653 C9PLK4 45263610 IC50 > 2000 nM T02653 C78JKD 45265930 IC50 = 1100 nM T02653 C08UBE 45272032 IC50 > 10000 nM T02653 C57EZH 45275745 IC50 = 110 nM T02653 CU7D0O 45278780 IC50 = 3.7 nM T02653 CY8A1D 45278857 IC50 = 3.1 nM T02653 CGX87F 45279098 IC50 = 6.5 nM T02653 CL9P2A 45380783 IC50 = 3.8 nM T02653 CKC0B7 46237842 IC50 = 59 nM T02653 C4KN0J 46237981 IC50 = 31 nM T02653 C7KW8T 46883839 EC50 > 10000 nM T02653 CZSG25 46883893 EC50 > 10000 nM T02653 C72MUY 46889765 IC50 > 5000 nM T02653 C6DVO1 46889848 IC50 > 10000 nM T02653 CZ90FC 46894119 Ki = 9 nM T02653 C04KWS 46913888 IC50 = 54 nM T02653 C1U7QL 46913889 IC50 = 52 nM T02653 C3Q7RI 46913890 IC50 = 6 nM T02653 CY7D0I 46913891 IC50 = 80 nM T02653 CQ93ML 46913892 IC50 = 135 nM T02653 C1ZRD2 46914168 IC50 = 1620 nM T02653 CWV42M 46914169 IC50 = 3740 nM T02653 CK6SJ3 46914453 IC50 = 275 nM T02653 C4HQ5Y 46914584 IC50 = 223 nM T02653 C9F4PR 46914585 IC50 = 4340 nM T02653 CZE49A 46914586 IC50 = 553 nM T02653 CGS9U8 46914587 IC50 = 41 nM T02653 C34EDY 46914588 IC50 = 21 nM T02653 CLCI21 46914734 IC50 = 13 nM T02653 C2NM6E 46914737 IC50 = 25 nM T02653 CKP01L 46914738 IC50 = 58 nM T02653 CP91XE 46914741 IC50 = 89 nM T02653 C3Q5PE 46914742 IC50 = 4 nM T02653 C6OG0A 46914743 IC50 = 7 nM T02653 C1TMA8 46914744 IC50 = 150 nM T02653 CE7KZ8 46914881 IC50 = 83 nM T02653 CI0Y4F 46914882 IC50 > 10000 nM T02653 C8HWO7 46914883 IC50 = 784 nM T02653 C6FN4G 46914884 IC50 = 246 nM T02653 CXY74T 46914885 IC50 = 9730 nM T02653 CF1D5Q 46914886 IC50 = 488 nM T02653 CVGF35 46914887 IC50 > 500 nM T02653 C4ZPR6 46915029 IC50 = 180 nM T02653 CXR29C 46915030 IC50 > 10000 nM T02653 C9NC0K 46915031 IC50 = 1440 nM T02653 CY3O2C 46915043 IC50 = 41 nM T02653 CHG94E 46915044 IC50 = 32 nM T02653 CK85FJ 46915045 IC50 = 101 nM T02653 CQ6J3N 46915201 IC50 = 2080 nM T02653 CC84WO 46915202 IC50 = 8360 nM T02653 CTM2J5 46915203 IC50 = 31 nM T02653 C75IFZ 46915353 IC50 = 16 nM T02653 CJW51A 46915354 IC50 = 26 nM T02653 CX70GY 46915355 IC50 = 15.2 nM T02653 CPTL45 46915356 IC50 = 2 nM T02653 C39SUV 46915640 IC50 = 243 nM T02653 CX6WK5 46915641 IC50 = 535 nM T02653 CW8J2E 46915642 IC50 = 56 nM T02653 C05YTF 46915643 IC50 = 284 nM T02653 CMW7E4 46915644 IC50 = 56 nM T02653 CA43UG 46915645 IC50 > 127 nM T02653 CJ3DN2 46915781 IC50 > 1000 nM T02653 C4L1JF 46915782 IC50 = 383 nM T02653 CB4X3D 46915783 IC50 > 10000 nM T02653 CK7DI0 46915784 IC50 > 10000 nM T02653 CU7L4T 46915785 IC50 = 10000 nM T02653 CE9OU3 46915786 IC50 = 410 nM T02653 CI3E2M 46915787 IC50 = 763 nM T02653 C1BV5K 46916070 IC50 = 3650 nM T02653 C06JHQ 46916071 IC50 = 441 nM T02653 CQ37UY 46916072 IC50 = 1590 nM T02653 C38HIP 46916073 IC50 = 1290 nM T02653 CPK95L 46916074 IC50 = 151 nM T02653 C7NC4B 46917090 IC50 = 2.8 nM T02653 C2LCJ7 46937290 IC50 = 210 nM T02653 CKQ8J3 46937431 IC50 > 2000 nM T02653 CL7P3N 46938234 IC50 = 1.8 nM T02653 COS28G 46938235 IC50 = 18 nM T02653 CFJT93 46938236 IC50 = 7.6 nM T02653 CHL70M 46938239 IC50 = 4.1 nM T02653 C8P7JH 46938914 IC50 > 2000 nM T02653 CY95VK 46938915 IC50 > 2000 nM T02653 CVX25Q 46938916 IC50 = 220 nM T02653 C2V5AT 46939019 IC50 = 480 nM T02653 C5R6GI 46939020 IC50 = 390 nM T02653 CF1BX0 46939115 IC50 > 2000 nM T02653 C4P0EU 46939116 IC50 = 160 nM T02653 CD6B7X 46939395 IC50 = 58 nM T02653 C1KXF2 46939396 IC50 > 2000 nM T02653 CVN4W1 47958757 IC50 = 168 nM T02653 CX0NO8 49782554 EC50 < 15848.93 nM T02653 CC7T8Q 49782555 EC50 < 15848.93 nM T02653 CD07EV 49782777 EC50 < 15848.93 nM T02653 C43UKW 49782778 IC50 < 14421.15 nM T02653 C2JTF0 49782779 EC50 < 15848.93 nM T02653 CS7KX9 49782780 IC50 < 12560.3 nM T02653 C36RYU 49782781 IC50 = 5140.44 nM T02653 C8OA0C 49782985 EC50 < 15848.93 nM T02653 C5Y6QU 49782986 EC50 < 15848.93 nM T02653 CB8V7R 49782987 EC50 < 15848.93 nM T02653 CU3S6H 49836028 EC50 > 5000 nM T02653 C96SLW 49851364 EC50 > 5000 nM T02653 CDN4K6 49851369 EC50 > 5000 nM T02653 C4YXN1 49851467 EC50 > 5000 nM T02653 CUD91T 49862248 EC50 > 10000 nM T02653 C5NX4D 49864061 IC50 = 2530 nM T02653 CPH9D8 49864098 IC50 = 69 nM T02653 CMS1N3 49864127 IC50 = 15 nM T02653 CTE0N7 49864128 IC50 = 720 nM T02653 COP7W2 49864129 IC50 = 127 nM T02653 CCKJ45 49864153 IC50 = 849 nM T02653 C19FRV 49864154 IC50 = 65 nM T02653 CWGD27 49864174 IC50 = 146 nM T02653 C9YCN1 49864175 IC50 = 39 nM T02653 CTKV39 49864176 IC50 = 26 nM T02653 CZ8J1V 50942115 Ki = 800 nM T02653 C23OEF 50942312 EC50 > 10000 nM T02653 CX1KO8 51346768 Ki = 849 nM T02653 C7N9TD 51346823 Ki = 1518 nM T02653 C0WDX3 51347001 Ki = 1115 nM T02653 CF8DK7 51347002 Ki = 3170 nM T02653 CTH45Q 52918523 IC50 > 10000 nM T02653 CL8D1Z 52921432 IC50 = 130 nM T02653 CEC4I7 52941608 IC50 = 230 nM T02653 CDV90J 52942528 IC50 > 1000 nM T02653 C8Y9SU 52944898 IC50 > 1000 nM T02653 CK5UT4 53317489 Ki = 126 nM T02653 CM0LU1 53318659 Ki = 1200 nM T02653 CUD48O 53320087 Ki = 0.64 nM T02653 CD0N1K 53323476 IC50 = 356 nM T02653 CYH3V0 53325642 Ki = 86.8 nM T02653 C82DYI 53326614 Ki > 4170 nM T02653 CJCP75 53359074 EC50 > 5000 nM T02653 C9H5YE 53361128 EC50 > 5000 nM T02653 CUR24K 53875787 IC50 = 2800 nM T02653 C1JR5W 54576068 IC50 = 24 nM T02653 CS62XZ 54590901 IC50 = 53.9 nM T02653 C30XLO 54592009 Ki = 6.3 nM T02653 CCS8R6 54592010 IC50 = 39 nM T02653 CML2E7 54592011 IC50 = 86 nM T02653 CRVB01 54592087 IC50 = 266 nM T02653 C7W1BA 54592088 IC50 = 109 nM T02653 C9N3IS 54592089 IC50 = 56 nM T02653 C2GML6 54592090 IC50 = 33 nM T02653 C05FVP 54592092 IC50 = 19 nM T02653 C9W5DZ 56593984 EC50 > 5000 nM T02653 CF3G2M 56925477 IC50 = 36 nM T02653 CZ7O8G 56925478 IC50 = 69 nM T02653 CV5C0T 56925479 IC50 > 10000 nM T02653 C9ITY0 56925480 IC50 > 10000 nM T02653 C3M4TE 56925570 IC50 = 920 nM T02653 CZ4I2J 56925571 IC50 = 6800 nM T02653 CW87RG 56925573 IC50 = 2000 nM T02653 C4Z5LF 56925574 IC50 = 4100 nM T02653 CKF8Z3 56925575 IC50 = 1300 nM T02653 CY20OR 56925668 IC50 > 10000 nM T02653 C30DAL 56925669 IC50 = 600 nM T02653 CQHA65 56925670 IC50 = 310 nM T02653 CJP31U 56925671 IC50 = 270 nM T02653 CV86DS 56925673 IC50 = 2700 nM T02653 CI3S6F 56925790 IC50 = 5300 nM T02653 CTY1Q9 56925791 IC50 = 1100 nM T02653 CH40YG 56925792 IC50 = 960 nM T02653 C2PLD4 56925793 IC50 = 260 nM T02653 CU02HT 56925794 IC50 = 570 nM T02653 CM19WI 56925904 IC50 > 10000 nM T02653 CA7BX4 56925905 IC50 = 440 nM T02653 CTR7X3 56925906 IC50 = 1100 nM T02653 C39VBK 56925907 IC50 = 430 nM T02653 CV7EN5 56925908 IC50 = 320 nM T02653 CU69SK 56925909 IC50 = 590 nM T02653 CAMI87 56925910 IC50 = 700 nM T02653 CTG9I7 56926011 IC50 = 70 nM T02653 CPD82H 56968080 IC50 = 7.1 nM T02653 CM0SG2 57390990 IC50 = 1100 nM T02653 CU8AN3 57392780 IC50 = 790 nM T02653 CX12JM 57392781 IC50 = 45 nM T02653 C9OMW1 57392782 IC50 = 405 nM T02653 C30JOV 57394501 IC50 = 190 nM T02653 CINU04 57396254 IC50 = 225 nM T02653 C1O6JU 57396255 IC50 = 230 nM T02653 CVOB64 57399718 IC50 = 610 nM T02653 CF83VM 57401459 EC50 > 5000 nM T02653 C7W3YD 57401479 IC50 = 430 nM T02653 CR6L7E 57403222 IC50 = 1450 nM T02653 CPU6W7 57473898 IC50 = 80 nM T02653 CEJ25K 57473899 IC50 = 270 nM T02653 CUJ08D 57474008 IC50 = 70 nM T02653 CDB0F1 57503322 IC50 = 39 nM T02653 CIDS61 57503325 IC50 = 19 nM T02653 C2U1GQ 57524309 IC50 = 22 nM T02653 C0BDS9 57585514 IC50 < 2 nM T02653 CM17UZ 57585515 IC50 = 47 nM T02653 CYGU85 57585534 IC50 = 1.3 nM T02653 C3WG0L 57666312 Ki = 1100 nM T02653 C43GDR 57666397 Ki = 290 nM T02653 CTM6K5 57690900 IC50 > 5000 nM T02653 CB2I7A 57748722 Ki <= 10 nM T02653 CT9Y6X 57748723 Ki <= 10 nM T02653 C6J0HD 57748748 Ki <= 10 nM T02653 C2MFH6 57748755 Ki <= 10 nM T02653 CMR56T 57748765 Ki <= 10 nM T02653 C05UIP 57748768 Ki <= 10 nM T02653 CH2PV6 57748780 Ki = 0.79 nM T02653 CL13HZ 57748781 Ki = 0.4 nM T02653 C7UH3N 57748789 Ki <= 10 nM T02653 C2YT7S 57748790 Ki = 0.23 nM T02653 C1KZT3 57906156 IC50 = 500 nM T02653 C3IN9F 57983276 IC50 = 170 nM T02653 CJ6Y1B 58026134 IC50 > 2000 nM T02653 C19XQV 58026164 IC50 > 2000 nM T02653 CR7H3O 58026170 IC50 > 2000 nM T02653 C7XL3D 58026176 IC50 > 2000 nM T02653 CT1EM3 58064710 IC50 = 3.7 nM T02653 C8S3EQ 58064714 IC50 = 2.7 nM T02653 CPI62D 58064720 IC50 = 2.2 nM T02653 CL42XF 58064726 IC50 = 4.3 nM T02653 CPL9A6 58064729 IC50 = 55.9 nM T02653 CRFS78 58064730 IC50 = 3.3 nM T02653 CN1J3V 58064734 IC50 = 17.8 nM T02653 CA0SH5 58064735 IC50 = 4.4 nM T02653 CI7BP4 58064741 IC50 = 21.4 nM T02653 C2FZA7 58064756 IC50 = 9.4 nM T02653 C3AMO0 58064757 IC50 = 4450 nM T02653 C47AUR 58392644 EC50 = 2.5 nM T02653 C9CQS0 58392665 EC50 = 3.2 nM T02653 CXF39M 58392685 EC50 > 3000 nM T02653 C7FXH3 58392721 EC50 > 3000 nM T02653 CJDN90 58392790 EC50 = 1.6 nM T02653 CO59DQ 58392803 EC50 > 3000 nM T02653 C5K9PJ 58483018 IC50 = 1.2 nM T02653 C4C2FT 58599563 IC50 = 1300 nM T02653 CWAD17 58731166 Ki <= 500 nM T02653 CNE02T 58731180 Ki <= 500 nM T02653 CVS58C 58731199 Ki <= 500 nM T02653 C3VU0Q 58731202 Ki <= 500 nM T02653 C03HFM 58731234 Ki <= 500 nM T02653 CADQ18 58731243 Ki <= 500 nM T02653 CI7XQ5 58731245 Ki <= 500 nM T02653 C67UET 58731323 Ki <= 500 nM T02653 C0JL7A 58973277 IC50 > 1000 nM T02653 CY38HG 59233337 Ki > 1000 nM T02653 CUX4E7 59233347 Ki > 3333 nM T02653 CO63VJ 59233364 Ki > 1000 nM T02653 C2A9JO 59251119 IC50 > 5000 nM T02653 CD8A6P 59281281 IC50 = 49 nM T02653 CBZ0M5 59281312 IC50 = 170 nM T02653 CCT59B 59281329 IC50 = 510 nM T02653 CQI5C4 59281343 IC50 = 38 nM T02653 CH5E1F 59281346 IC50 > 10000 nM T02653 CPE83R 59281354 IC50 = 180 nM T02653 CI9EP1 59281363 IC50 = 8.4 nM T02653 CQ2BO1 59281403 IC50 = 51 nM T02653 CP78RD 59281411 IC50 = 95 nM T02653 CCNU12 59281412 IC50 = 10 nM T02653 C7HVB1 59281416 IC50 = 490 nM T02653 CE5A0V 59281447 IC50 = 75 nM T02653 CZT9S6 59281449 IC50 = 430 nM T02653 CIKQ89 59281508 IC50 = 990 nM T02653 CE1A7J 59281531 IC50 = 680 nM T02653 CK9JZ4 59281538 IC50 = 36 nM T02653 C4TG5U 59281540 IC50 = 22 nM T02653 CPC80S 59281541 IC50 = 64 nM T02653 CXS5C4 59281543 IC50 = 250 nM T02653 C7KPR9 59281566 IC50 = 150 nM T02653 CUJP64 59281599 IC50 = 600 nM T02653 CYZI85 59556974 IC50 > 10000 nM T02653 C5C3AO 59770003 Ki = 2.48 nM T02653 CH36PL 59807625 IC50 < 500 nM T02653 C54ATL 59807726 IC50 < 500 nM T02653 C8S7OB 59808080 IC50 < 500 nM T02653 CYU57B 59808129 IC50 < 500 nM T02653 C2TNO8 60026286 IC50 > 2000 nM T02653 CZE5J8 60026377 IC50 > 2000 nM T02653 C0LDS2 60026592 IC50 = 1150 nM T02653 C31PTC 60026641 IC50 > 2000 nM T02653 C67NSE 60026675 IC50 > 2000 nM T02653 C6GP5R 60026731 IC50 = 720 nM T02653 C5M8HV 60026772 IC50 = 1200 nM T02653 CI36XS 60026787 IC50 > 2000 nM T02653 C3JD8M 60026802 IC50 > 2000 nM T02653 CE9MI4 60026817 IC50 = 1900 nM T02653 C04EKW 60026878 IC50 > 2000 nM T02653 CPRW14 66991384 IC50 = 160 nM T02653 CYP31Z 66995780 IC50 = 3050 nM T02653 CK36QI 66996020 IC50 > 10000 nM T02653 CJ09TZ 66996063 IC50 = 2225 nM T02653 C3EU7N 66996137 IC50 = 276 nM T02653 C1CXY9 66996546 IC50 = 401 nM T02653 C9Y2DN 66996560 IC50 = 727 nM T02653 C9LOZ1 66996568 IC50 = 1181 nM T02653 CH39DP 67053383 IC50 > 2000 nM T02653 C3LF8O 67053425 IC50 > 2000 nM T02653 CMYP75 67415874 IC50 = 100 nM T02653 CQU8E3 68031408 IC50 = 11 nM T02653 C1FK3D 69081573 IC50 = 31 nM T02653 CB6HX8 69082589 IC50 = 480 nM T02653 C43PON 69675755 IC50 = 9.4 nM T02653 COR52G 69675880 IC50 = 13 nM T02653 C9Q7VH 70561849 IC50 = 39 nM T02653 CARO49 70685018 Ki = 150 nM T02653 C5QPC0 70697572 Ki = 170 nM T02653 C94FCP 71452686 IC50 = 3000 nM T02653 CF08ME 71457470 Ki = 0.4 nM T02653 CEO5G4 71461616 IC50 = 1900 nM T02653 C78IOK 71467161 IC50 = 310 nM T02653 C1MHC0 71467246 IC50 = 47 nM T02653 C4B0IC 71467248 IC50 = 26 nM T02653 CYW34A 71519686 IC50 = 120 nM T02653 CGK4S8 71543393 Ki = 1450 nM T02653 C83YJF 71544946 IC50 = 39 nM T02653 CK2O1Z 71545110 IC50 = 54 nM T02653 C0LD8K 71548690 IC50 = 270 nM T02653 C19CGP 71548691 IC50 = 1700 nM T02653 C4BE6G 71548692 IC50 = 1110 nM T02653 CCK7Q3 71548693 IC50 = 240 nM T02653 CK9S0J 71548694 IC50 = 1440 nM T02653 CT9Y5D 71549558 Ki = 2 nM T02653 C8ZX0F 71549573 IC50 = 180 nM T02653 COQ5C4 71549690 IC50 = 230 nM T02653 CE7NZ0 71549691 IC50 = 190 nM T02653 C1ZF5V 71549692 IC50 = 180 nM T02653 C15JLF 71549694 IC50 = 120 nM T02653 CUX57Y 71549702 IC50 = 200 nM T02653 CQX42S 71549703 IC50 = 190 nM T02653 CZ3C8X 71549705 IC50 = 500 nM T02653 C0IH6J 71549706 IC50 = 170 nM T02653 CZ8Y7O 71549829 IC50 = 40 nM T02653 CPS61I 71549840 IC50 = 37 nM T02653 CC5AU3 71549841 IC50 = 55 nM T02653 CCV90M 71549842 IC50 = 14 nM T02653 CPFL57 71549843 IC50 = 33 nM T02653 CY8SP0 71549969 IC50 = 210 nM T02653 CXP57U 71549980 IC50 = 180 nM T02653 CA64KN 71550109 IC50 = 400 nM T02653 CUG9C6 71550110 IC50 = 30 nM T02653 CK7NS4 71550116 IC50 = 270 nM T02653 COW8K4 71550118 IC50 = 340 nM T02653 C50TXO 71550241 IC50 = 33 nM T02653 CX6JR5 71550242 IC50 = 34 nM T02653 C93KZM 71550243 IC50 = 42 nM T02653 C6WIA2 71550244 IC50 = 120 nM T02653 CX26UJ 71550250 IC50 = 990 nM T02653 C7R1LJ 71550386 IC50 = 800 nM T02653 CMVD92 71550387 IC50 = 150 nM T02653 CUK7A8 71550511 IC50 = 160 nM T02653 CYB2L0 71550527 IC50 = 230 nM T02653 C6XF9J 71550528 IC50 = 370 nM T02653 CJYQ15 71550529 IC50 = 170 nM T02653 CSHT69 71550657 IC50 = 82 nM T02653 CJX19L 71550659 IC50 = 1530 nM T02653 C6SNW1 71550660 IC50 = 130 nM T02653 CU0Q9P 71550799 IC50 = 470 nM T02653 C8SDX6 71550801 IC50 = 68 nM T02653 CK3HZ0 71550802 IC50 = 240 nM T02653 C9QD8V 71726436 IC50 = 300 nM T02653 CKO01U 71726437 IC50 > 40000 nM T02653 CP9M2C 71726438 IC50 = 750 nM T02653 C6TXD3 71726439 IC50 = 450 nM T02653 CP62QW 71726440 IC50 > 40000 nM T02653 CQYH84 71726556 IC50 > 40000 nM T02653 C8N4UF 71726557 IC50 > 40000 nM T02653 C6TXF5 71726558 IC50 = 500 nM T02653 C4RY0L 71726559 IC50 = 400 nM T02653 CPL35F 71726560 IC50 = 2900 nM T02653 C07YPM 71726687 IC50 > 40000 nM T02653 C6OQT5 71726688 IC50 > 40000 nM T02653 C7F3PL 71726689 IC50 > 40000 nM T02653 C91RTU 71726690 IC50 > 40000 nM T02653 CAR9T3 71726691 IC50 > 40000 nM T02653 C1E3QT 71726810 IC50 > 10000 nM T02653 CV02SB 71726811 IC50 > 40000 nM T02653 C0OXK4 71726812 IC50 > 40000 nM T02653 CL8Z2I 71726813 IC50 = 250 nM T02653 CWS86Q 71726934 IC50 = 3000 nM T02653 C62XFJ 71726935 IC50 > 10000 nM T02653 CIR49D 71726936 IC50 > 40000 nM T02653 CMO7T2 71726937 IC50 = 13000 nM T02653 CE67IF 71726938 IC50 = 16000 nM T02653 CEI4R9 71726939 IC50 > 40000 nM T02653 CKFV04 71727059 IC50 = 2500 nM T02653 CEK6Y8 71727060 IC50 = 1500 nM T02653 CJ0Z6D 71727061 IC50 = 3000 nM T02653 CAG0M9 71727062 IC50 = 300 nM T02653 CN4TI1 71727063 IC50 = 4000 nM T02653 CB45XH 71727183 IC50 = 15000 nM T02653 C76QBF 71727184 IC50 > 40000 nM T02653 CIY4W8 71727185 IC50 > 40000 nM T02653 CB12CL 71727731 IC50 = 6000 nM T02653 C91POE 71727732 IC50 = 1000 nM T02653 C6O2YB 71727733 IC50 = 300 nM T02653 CIUT23 71727734 IC50 = 1000 nM T02653 CE6GH7 71727735 IC50 = 500 nM T02653 CDME45 71727852 IC50 = 3000 nM T02653 C8W7UV 71727853 IC50 = 200 nM T02653 CLTX21 71727854 IC50 = 280 nM T02653 CG0Y6I 71727855 IC50 = 400 nM T02653 C6A1KB 71727856 IC50 = 2600 nM T02653 CRS9A7 71727980 IC50 = 570 nM T02653 CRC7E9 71727981 IC50 = 500 nM T02653 CCK75S 71727982 IC50 > 10000 nM T02653 C3X0QV 71727983 IC50 = 3000 nM T02653 C2KIM1 71727984 IC50 = 600 nM T02653 CKQN54 71728108 IC50 = 2000 nM T02653 C2W9HE 71728109 IC50 = 1000 nM T02653 CVL7Q6 71728110 IC50 = 100 nM T02653 CM78AL 71728111 IC50 = 300 nM T02653 CN80TQ 71728112 IC50 = 100 nM T02653 CF52OE 71728113 IC50 = 4000 nM T02653 C8BGF3 71728224 IC50 = 1200 nM T02653 CJ4M6P 71728225 IC50 = 2000 nM T02653 C10AOX 71728227 IC50 > 30000 nM T02653 C4XSM7 71728228 IC50 = 3000 nM T02653 CW5C6N 71728229 IC50 = 280 nM T02653 CP5KM8 72163477 IC50 = 660 nM T02653 CA6O4K 72163478 IC50 = 750 nM T02653 C27XWS 72163479 IC50 = 1200 nM T02653 C6M9CN 72163480 IC50 = 120 nM T02653 CL8AH4 72163481 IC50 = 550 nM T02653 CB2SD9 72163621 IC50 = 1200 nM T02653 CU6NA8 72163622 IC50 = 170 nM T02653 CTEV75 72163623 IC50 = 33 nM T02653 CER73F 72163624 IC50 = 68 nM T02653 CC8VM7 72163625 IC50 = 1600 nM T02653 CS69AC 72163626 IC50 = 94 nM T02653 CAJ0H5 72163627 IC50 = 43 nM T02653 C1D3EU 72163754 IC50 = 92 nM T02653 C1G3ES 72163755 IC50 = 23 nM T02653 CP8AC2 72188914 EC50 > 5000000 nM T02653 CA6FO5 72188915 EC50 > 5000000 nM T02653 CZ5O6M 72204151 IC50 = 3500 nM T02653 CGT02E 72204156 IC50 = 10900 nM T02653 CW6I9L 72204538 EC50 = 4100 nM T02653 CH5Q8D 72544150 IC50 = 40 nM T02653 C4YUD1 72544151 IC50 = 45 nM T02653 CTM6Y0 72544152 IC50 = 2029 nM T02653 C2K7JR 72544153 IC50 = 1393 nM T02653 C0ZGC8 72544374 IC50 = 1530 nM T02653 CC64LQ 72544375 IC50 = 1974 nM T02653 CNG1C6 72544376 IC50 = 4698 nM T02653 CS1QT2 72544377 IC50 = 121 nM T02653 C0X6YV 72544378 IC50 = 1207 nM T02653 C97CRH 72544379 IC50 = 342 nM T02653 CJ8N2H 72544380 IC50 = 1844 nM T02653 CRB36F 72544601 IC50 = 2086 nM T02653 C3LJ6V 72544602 IC50 = 627 nM T02653 C34FBN 72544603 Ki = 113 nM T02653 CLA3Y9 72710581 Ki = 6.1 nM T02653 CXB45U 72724690 IC50 = 270 nM T02653 CI2K6C 72725442 IC50 = 700 nM T02653 C0W2UD 72725443 IC50 = 400 nM T02653 CQ5D1B 72725444 IC50 = 1100 nM T02653 C2PJV7 72725445 IC50 > 10000 nM T02653 CQ4Z2C 72725446 IC50 = 350 nM T02653 C47IMQ 72725447 IC50 = 2400 nM T02653 CJSK52 72725491 IC50 = 360 nM T02653 CS6J4T 72725492 IC50 = 400 nM T02653 C41FYD 72725493 IC50 = 150 nM T02653 CUG96L 72725494 IC50 = 190 nM T02653 CFHJ16 72725495 IC50 = 400 nM T02653 CW7IY3 72725496 IC50 = 330 nM T02653 CSV1I7 72725497 IC50 = 240 nM T02653 COV09R 72725548 IC50 = 320 nM T02653 CTE01I 72725549 IC50 = 1400 nM T02653 C09ZFS 72725550 IC50 = 480 nM T02653 C2Z7QT 72725551 IC50 = 110 nM T02653 C0K2CP 72725552 IC50 = 5200 nM T02653 C37MEN 72725553 IC50 = 1000 nM T02653 CYSM01 72725554 IC50 = 2300 nM T02653 COU49R 76314656 IC50 = 170 nM T02653 C95NBT 76314657 IC50 > 2000 nM T02653 CL95NP 76317025 IC50 = 609 nM T02653 CZ08OF 76317198 IC50 = 510 nM T02653 CR5B2V 76317199 IC50 = 470 nM T02653 C5YFZ6 76318225 IC50 > 2000 nM T02653 C0RK5D 76321918 IC50 = 1100 nM T02653 C3IC5B 76329113 IC50 > 2000 nM T02653 C1RB6X 76329114 IC50 = 260 nM T02653 CP8M1Z 76332766 IC50 > 2000 nM T02653 CKDI18 76332767 IC50 > 2000 nM T02653 CK21EY 77461202 IC50 = 420 nM T02653 CX20VN 84429708 Ki = 1000 nM T02653 CIU65X 86280440 Ki = 1580 nM T02653 CH46CP 87361539 Ki = 0.08 nM T02653 CT50AL 87539277 IC50 > 1000 nM T02653 CY05IC 87733533 IC50 > 1000 nM T02653 C9EH7I 89500376 Ki > 7010 nM T02653 C0EQS7 89501406 Ki = 415 nM T02653 CG67BU 89508836 IC50 = 130 nM T02653 CBLU18 89509944 IC50 = 380 nM T02653 C8JG7O 89510193 Ki = 1840 nM T02653 CK5D1A 90395281 IC50 = 220 nM T02653 CPC47K 90396922 IC50 = 1600 nM T02653 CQ06RH 90654508 IC50 = 1300 nM T02653 CY5L7N 90655674 IC50 = 660 nM T02653 C9B0QF 90655675 IC50 = 1320 nM T02653 CG6QP2 90655676 IC50 = 670 nM T02653 C8EH0K 90655677 IC50 = 6740 nM T02653 C8GQ4S 90655678 IC50 = 270 nM T02653 C6VZ7X 90656360 IC50 = 9 nM T02653 CNCB43 90656361 IC50 = 10.7 nM T02653 CS42NY 90656362 IC50 = 30.7 nM T02653 C2ZF7W 110763791 Ki = 630.96 nM T02653 CD7RS9 118599615 Ki = 3.981 nM T02653 C70AOV 118599714 Ki = 63.1 nM T02653 C8XLO9 118599727 EC50 = 12.59 nM T02653 CYCM67 118599740 IC50 > 10000 nM T02653 CW7G4T 118599742 Ki = 2.512 nM T02653 C9L5EW 118599756 Ki = 158.49 nM T02653 CVIW94 118599769 EC50 = 1 nM T02653 CFS28Y 118599779 Ki = 50.12 nM T02653 CLS7C1 118707978 EC50 > 5000 nM T02653 C9LV0M 118707979 EC50 > 5000 nM T02653 CC2H4E 118714881 IC50 = 710 nM T02653 C2MQ3P 118714882 IC50 > 10000 nM T02653 CE3I9T 118723172 IC50 > 2000 nM T02653 C13AIC 118723173 IC50 > 2000 nM T02653 C21SWI 118723174 IC50 > 2000 nM T02653 CKR24J 118723175 IC50 > 2000 nM T02653 C28YZF 118723176 IC50 > 2000 nM T02653 C6AGI7 118723177 IC50 > 2000 nM T02653 C4QO8E 118723178 IC50 > 2000 nM T02653 C1RYW9 118796369 Ki = 2 nM T02653 C0X8SA 122178358 IC50 = 1200 nM T02653 C14KFA 122178359 IC50 = 420 nM T02653 C04DIU 122178360 IC50 = 62 nM T02653 CG13LX 122178361 IC50 = 39 nM T02653 C40DRP 122178362 IC50 = 120 nM T02653 C6IV5P 122178363 IC50 = 36 nM T02653 C3MLD0 122178364 IC50 = 64 nM T02653 C0NEZ7 122178365 IC50 = 72 nM T02653 CIT71M 122178366 IC50 = 150 nM T02653 C5ON0U 122178367 IC50 = 1100 nM T02653 C9LIR4 122179356 Ki = 337 nM T02653 CUI57B 122179357 Ki > 3000 nM T02653 CY18QG 122186737 Ki = 2120 nM T02653 C0OR2H 122186738 Ki = 6530 nM T02653 CU0Y8B 122186739 Ki = 3890 nM T02653 CWF0Q4 122186740 Ki = 38.4 nM T02653 CBE6Q8 122186741 Ki = 3880 nM T02653 CX13DR 122186742 Ki = 4250 nM T02653 CJ74HX 122186743 Ki = 3920 nM T02653 C05VWL 122186744 Ki = 44.7 nM T02653 CNX5H4 122186745 Ki = 4470 nM T02653 CQ6BG8 122186747 Ki = 2.1 nM T02653 CH8O2M 122186748 Ki = 27.4 nM T02653 C4LRN1 122186749 Ki = 225 nM T02653 CCK36V 127029882 Ki = 6 nM T02653 CVC84H 127029883 Ki = 6 nM T02653 CFY1P0 127029884 Ki = 6 nM T02653 CU1S6C 127029885 Ki = 7 nM T02653 CA1J0H 127030193 Ki = 1080 nM T02653 CU8Y7N 127030224 Ki = 31 nM T02653 CTEA14 127030225 IC50 = 56 nM T02653 CQ74CG 127030810 Ki = 162 nM T02653 CS5JP0 127031149 Ki = 694 nM T02653 CBW17G 127031150 Ki = 13 nM T02653 C19DUV 127031151 Ki = 14 nM T02653 CLDC46 127031152 Ki = 19 nM T02653 C60SMC 127031153 Ki = 16 nM T02653 C21UAK 127032030 Ki = 144 nM T02653 CBT43F 127032031 Ki = 258 nM T02653 C8TG9C 127032032 Ki = 980 nM T02653 CKZ3X7 127032033 Ki = 55 nM T02653 C8SOU3 127032034 Ki = 230 nM T02653 C87NBI 127032035 Ki = 1452 nM T02653 CKA18M 127032339 Ki > 10 nM T02653 CBR31K 127033260 Ki = 20 nM T02653 CAN7K2 127034410 IC50 = 5217 nM T02653 CSC7I2 127034411 Ki = 1092 nM T02653 C9TG2N 134137487 IC50 > 1000 nM T02653 CTF0J3 135567449 Ki = 1.995 nM T02653 CN24YZ 135567451 EC50 = 0.05012 nM T02653 CPF3B4 135567452 Ki = 0.631 nM T02653 C5MXO2 136000568 Ki > 10000 nM T02653 CM6OX5 136000656 Ki = 2700 nM T02653 CZ2D6U 136059148 Ki = 1600 nM T02653 C6HOU3 136059149 Ki = 1040 nM T02653 CE1G9O 136059150 Ki = 1700 nM T02653 C7LSN6 136088946 Ki = 2800 nM T02653 C3SE8T 136216705 IC50 = 700 nM T02653 CZXM35 136216706 IC50 = 900 nM T02653 CX8H9R 137632028 IC50 = 3900 nM T02653 C0XZC3 137633972 IC50 = 1400 nM T02653 COI80Z 137634236 IC50 > 1000 nM T02653 CP2C7M 137635745 IC50 = 55 nM T02653 CPD87Y 137639726 IC50 > 1000 nM T02653 C3K6DU 137640356 IC50 = 4600 nM T02653 CHTB16 137642739 IC50 = 900 nM T02653 C7KIR1 137643684 IC50 = 6.2 nM T02653 C0J8FI 137646168 IC50 = 4800 nM T02653 CPNB08 137646648 Ki = 195.7 nM T02653 C30ZJF 137648477 IC50 > 1000 nM T02653 C7IG3B 137649694 IC50 = 25 nM T02653 CX63RY 137650280 IC50 = 900 nM T02653 CXWF54 137652695 IC50 = 1100 nM T02653 C69ECN 137653076 IC50 = 18 nM T02653 C8OP2T 137653676 IC50 = 2200 nM T02653 CO92KL 137654415 IC50 > 1000 nM T02653 C8PR9K 137654628 IC50 = 33.4 nM T02653 CX65AR 137656053 IC50 = 1400 nM T02653 CS29XF 137656107 Ki <= 10 nM T02653 C0PL8V 137658165 IC50 = 7 nM T02653 C9GQB2 137658303 IC50 = 1600 nM T02653 C5T7IK 147930449 Ki = 3.981 nM T02653 CCDV87 155511242 IC50 = 114 nM T02653 C28RHM 155514304 Ki = 125.89 nM T02653 CE2YJ9 155514399 Ki = 10 nM T02653 CQF09V 155516050 Ki = 50.12 nM T02653 CQ2GH0 155517818 IC50 = 6309.57 nM T02653 CELU49 155517819 IC50 > 10000 nM T02653 C2E4XV 155518137 Ki = 1000 nM T02653 C4QAB0 155518139 Ki = 1258.93 nM T02653 CCO0Z4 155519877 Ki = 10 nM T02653 C8BD6Y 155522508 Ki = 12.59 nM T02653 CILC13 155524288 IC50 = 5940 nM T02653 C71VIK 155525344 EC50 = 12.59 nM T02653 C1WAQ6 155527406 Ki = 199.53 nM T02653 C5T2QN 155528866 IC50 = 100 nM T02653 CBO7E4 155528935 Ki = 501.19 nM T02653 CQM89D 155529443 Ki < 0.3162 nM T02653 CR0N3F 155529454 Ki = 7.943 nM T02653 CB0XS4 155529625 IC50 > 10000 nM T02653 CLC65H 155532000 Ki = 1995.26 nM T02653 C3HFZ6 155534085 IC50 > 10000 nM T02653 CF52DM 155535034 Ki = 0.5012 nM T02653 CXR2W1 155536089 IC50 = 22 nM T02653 C3FON4 155537084 Ki = 398.11 nM T02653 CUI53F 155537601 Ki = 794.33 nM T02653 C78ISM 155540009 IC50 = 567 nM T02653 CIAW80 155544156 IC50 = 21990 nM T02653 C76OVS 155544396 Ki = 1000 nM T02653 CR6UY8 155545121 IC50 = 20 nM T02653 CE3VY8 155550102 Ki = 6309.57 nM T02653 C6H2ML 155552723 Ki = 7.943 nM T02653 CW8BH4 155554673 Ki = 39.81 nM T02653 C9WV3L 155556878 Ki = 15.85 nM T02653 CR5ZI2 155557239 IC50 = 63.1 nM T02653 CPY83L 155558503 IC50 > 10000 nM T02653 CFAN82 155561077 Ki = 63.1 nM T02653 CQ7HG2 155561626 Ki = 3.162 nM T02653 CXQ23E 155562099 IC50 = 7690 nM T02653 CD4K6Z 155564467 Ki = 0.3162 nM T02653 CS25QB 155564604 IC50 = 32 nM T02653 C7YK6N 155565026 IC50 = 64 nM T02653 C4XJU2 155565054 Ki = 501.19 nM T02653 CPX2J5 155566857 Ki > 6309.57 nM T02653 C79WFJ 155567245 IC50 > 10000 nM T02653 CME1B7 155567676 Ki = 316.23 nM T02653 D00ZGW 46883841 EC50 > 10000 nM T02653 D01ETZ 261000 Ki = 0.54 nM T02653 D01NVD 46830196 EC50 > 19952.62 nM T02653 D04UDT 10407950 IC50 = 126 nM T02653 D07KWO 9823099 IC50 = 6300 nM T02653 D08KQM 24816375 Ki = 149 nM T02653 D09OKK 9951771 IC50 < 20 nM T02653 D0F1SS 44605900 IC50 > 3000000 nM T02653 D0G5OV 11543746 IC50 = 3700 nM T02653 D0M0RS 11560224 Ki > 1000 nM T02653 D0V4RZ 25113722 IC50 > 10000 nM T02653 D0XS0R 44433505 Ki = 124 nM T11448 D01AZG 5073 Ki = 10 nM T11448 D01JGV 441975 Ki = 8.2 nM T11448 D01JUF 5775 Ki = 1.7 nM T11448 D03MIR 3157 Ki = 729 nM T11448 D03SKR 2803 Ki = 3.8 nM T11448 D04JEE 4946 IC50 > 5011.87 nM T11448 D04PHC 5816 EC50 = 30.2 nM T11448 D05MBZ 129211 Ki = 13.4 nM T11448 D05ZIK 4205 Ki = 20 nM T11448 D06OFS 68712 Ki = 36.31 nM T11448 D07MOX 439260 Ki = 66 nM T11448 D09EBS 4636 Ki = 0.29 nM T11448 D0AE3X 2435 EC50 = 0.6166 nM T11448 D0B1IV 14969 Ki = 50.12 nM T11448 D0E9PK 4810 Ki = 150 nM T11448 D0G8NN 119570 Ki = 75.7 nM T11448 D0H3HM 60795 Ki = 100 nM T11448 D0H4JM 8969 Ki = 0.42 nM T11448 D0H7KF 5002 Ki > 1000 nM T11448 D0K0MW 30668 Ki = 4.365 nM T11448 D0MT0M 2216 Ki = 2.9 nM T11448 D0P9RF 5401 Ki = 549.54 nM T11448 D0R6RO 4184 Ki = 4.8 nM T11448 D0TR5X 3386 Ki = 6.31 nM T11448 D0U3DU 5311068 EC50 = 1.5 nM T11448 D0V4QS 135398745 Ki = 192 nM T11448 D0WV3U 4893 Ki = 210 nM T11448 D0Z1RV 135398737 Ki = 24 nM T11448 D04DJS 3682 IC50 = 0.5 nM T11448 D05LGX 213041 Ki = 7.244 nM T11448 D0F2ML 68602 IC50 = 3400 nM T11448 D0LI1C 44469321 IC50 > 10000 nM T11448 D0N1HW 5311200 Ki = 170 nM T11448 D00OWF 5280953 Ki = 2540 nM T11448 D01RAE 133079 Ki > 1600 nM T11448 D02LHR 33625 Ki = 2240 nM T11448 D02ZSU 9838763 EC50 < 10000 nM T11448 D03QMR 5685 Ki = 3.5 nM T11448 D05FYA 3035905 Ki = 125.89 nM T11448 D05OVC 71310 Ki = 1.2 nM T11448 D08OWQ 122295 Ki = 114 nM T11448 D0B1MJ 6918097 Ki = 900 nM T11448 D0BC6Q 9837551 Ki = 1.2 nM T11448 D0EE6L 3038495 Ki = 2.75 nM T11448 D0K9JP 9928332 Ki = 2.4 nM T11448 D0L5TJ 10527469 Ki = 94.9 nM T11448 D0N7LZ 126225 Ki = 24 nM T11448 D0O7DB 9904117 Ki = 104.71 nM T11448 D0Z3UP 216249 EC50 > 10000 nM T11448 C4JQ7T 2068 Ki > 20000 nM T11448 C9X3BF 4786 Ki = 275.42 nM T11448 C5H9CN 9287 Ki = 630.96 nM T11448 CW59CR 20179 Ki = 20.89 nM T11448 CL3T5Z 27013 Ki < 100 nM T11448 CPK89W 43260 Ki = 1445.44 nM T11448 C3JL8A 43405 Ki = 1200 nM T11448 CU86VK 54459 Ki = 7.079 nM T11448 C28VFY 60602 Ki = 530 nM T11448 C4X7HB 72016 Ki = 4.4 nM T11448 C2X7YN 114697 Ki = 1560 nM T11448 CKP25M 121881 Ki < 1000 nM T11448 CKR4N3 122065 Ki = 1811 nM T11448 C2H1VA 131829 EC50 = 2.818 nM T11448 CLK7P3 169713 IC50 > 10000 nM T11448 CF4V5Q 185076 EC50 = 1.202 nM T11448 CX39NY 188249 Ki = 180 nM T11448 CH6WT3 218362 EC50 = 1.175 nM T11448 CQ5Z8Y 294234 Ki = 5.37 nM T11448 CPI2C5 2775690 Ki = 1202 nM T11448 CAQ2J0 3034396 Ki = 4720 nM T11448 CS2Q1G 3045401 IC50 = 0.5495 nM T11448 CYP29S 3073596 Ki = 6760.83 nM T11448 CU4T6Q 3086326 EC50 = 2.344 nM T11448 C0YXV3 3676358 Ki > 10000 nM T11448 C39UDN 5312114 IC50 = 97 nM T11448 C3A1FO 6604789 Ki = 7943.28 nM T11448 C8ZBJ9 7059292 Ki = 3019.95 nM T11448 CHD32K 9794524 Ki = 31 nM T11448 C4K7ZJ 9795515 Ki = 4.9 nM T11448 C5Z2KM 9805944 Ki = 1 nM T11448 C1NQC6 9807658 IC50 = 360 nM T11448 C6RW9F 9813756 Ki = 549.54 nM T11448 CJ67XC 9815610 Ki = 254 nM T11448 C9PZN8 9815633 Ki = 27 nM T11448 C5A8UR 9815707 EC50 = 1.622 nM T11448 CXP87Y 9816063 Ki = 68 nM T11448 C1X0UA 9817256 EC50 = 3311.31 nM T11448 C6KJ7P 9827677 Ki = 1288 nM T11448 CQZ6I0 9828476 Ki = 275.42 nM T11448 CS3MA5 9837106 Ki = 224 nM T11448 C6PL3A 9837600 Ki = 1.6 nM T11448 CCQ9W3 9838192 Ki = 169.82 nM T11448 CBN06W 9839050 Ki = 126 nM T11448 CB7L9H 9846548 Ki = 8.8 nM T11448 CY2D5T 9851486 Ki = 602.56 nM T11448 CM13ZV 9856041 IC50 > 10000 nM T11448 CQ2L0J 9859437 Ki = 6 nM T11448 C6ERH9 9863540 Ki > 3000 nM T11448 CBSE45 9865178 Ki = 33.11 nM T11448 CWU30O 9879119 Ki = 97.72 nM T11448 CV2HW7 9883506 Ki = 23.8 nM T11448 C3DB5H 9884781 Ki = 249 nM T11448 CTAC24 9885114 Ki = 411 nM T11448 C8HS4Q 9895326 Ki = 354.81 nM T11448 CY1P7H 9895868 IC50 = 7.7 nM T11448 CFI97S 9904205 IC50 = 371.54 nM T11448 CK89GE 9904606 Ki = 85.11 nM T11448 CYWQ50 9906447 Ki > 10000 nM T11448 C7JFZ5 9906978 Ki = 2239 nM T11448 C32ZXG 9923679 Ki = 500 nM T11448 CBMI05 9926529 Ki = 131.83 nM T11448 C03ZFH 9931977 Ki = 872 nM T11448 C4L1GA 9934033 IC50 = 104 nM T11448 CNWR13 9944409 Ki = 44.67 nM T11448 CBM62P 9944467 Ki = 309.03 nM T11448 CUQ8I5 9947861 Ki < 7943.28 nM T11448 CQI54C 9950711 Ki = 954.99 nM T11448 CO2X8D 9951544 IC50 = 1.738 nM T11448 CUA8K5 9953974 Ki = 3000 nM T11448 CF1C5Q 9960497 Ki = 800 nM T11448 C3O9SC 9971924 Ki = 30.9 nM T11448 CFN50J 9978683 Ki > 5000 nM T11448 C2CM4Y 9990389 Ki = 3.981 nM T11448 CQL12P 10004545 Ki > 2000 nM T11448 C1XK9Y 10019102 IC50 = 3000 nM T11448 C52JBP 10028898 Ki = 9.3 nM T11448 C2EUY0 10035109 Ki > 10000 nM T11448 CW26VU 10036255 Ki = 51 nM T11448 C9IQK6 10036256 Ki = 51 nM T11448 C5MZ6I 10042547 Ki = 2570.4 nM T11448 C7D0GO 10044968 Ki = 840 nM T11448 CB82XU 10045088 Ki = 3100 nM T11448 C3MTF4 10045713 Ki = 715 nM T11448 CLE0M4 10056237 Ki = 0.39 nM T11448 CZ0U2N 10070896 Ki = 1400 nM T11448 CX5EA7 10081626 Ki = 12 nM T11448 CKA5F4 10084076 Ki = 92.8 nM T11448 C7J1UB 10101373 Ki = 52 nM T11448 CQ9O8W 10105615 IC50 = 379800 nM T11448 CA5H7K 10106205 Ki = 19 nM T11448 C54EYD 10108561 IC50 < 1000 nM T11448 COF5U3 10109188 Ki = 1100 nM T11448 C3N8JR 10123375 Ki = 1.35 nM T11448 C9XCB3 10132386 Ki = 2210 nM T11448 CE27RV 10135864 EC50 > 10000 nM T11448 CWON56 10176433 Ki = 34 nM T11448 CQOE78 10176715 Ki = 100 nM T11448 CRS5B6 10176999 Ki = 1.7 nM T11448 CNB56M 10177445 Ki = 1700 nM T11448 C64WSY 10198108 Ki = 7 nM T11448 CQ8HX2 10198135 Ki = 10 nM T11448 C7MKP9 10199335 Ki = 4466.84 nM T11448 CC2KV3 10214826 Ki = 510 nM T11448 CLY2B9 10220232 Ki = 25 nM T11448 CU2B9P 10221004 Ki = 1318.26 nM T11448 CX9YD5 10221005 Ki = 3890.45 nM T11448 CNHR93 10231050 IC50 = 390 nM T11448 CVF1E5 10246054 IC50 > 1000 nM T11448 C0LOA6 10251036 Ki = 960 nM T11448 C6FH4C 10262765 Ki = 12 nM T11448 C6G0AY 10266032 Ki = 15.14 nM T11448 C3ZJY6 10303307 IC50 = 570 nM T11448 CBE9K1 10317643 Ki = 1380 nM T11448 C4MD0S 10318507 Ki = 1430 nM T11448 CSU1R6 10319299 Ki = 1700 nM T11448 C3NGO6 10332138 Ki = 3400 nM T11448 C6W5DM 10333157 EC50 = 74.13 nM T11448 C3E5CB 10337773 Ki = 31622.78 nM T11448 C1A3KN 10350094 Ki = 1.73 nM T11448 CN8PA7 10357986 IC50 = 6200 nM T11448 COS13I 10362866 Ki = 1850 nM T11448 CS2DN8 10376336 IC50 = 61900 nM T11448 C4H6YF 10379435 Ki = 5623.41 nM T11448 CDAC63 10381889 IC50 = 478.63 nM T11448 C3N7TF 10382537 Ki = 6.761 nM T11448 CMZA83 10383646 Ki > 5000 nM T11448 CRK20B 10398419 Ki = 87 nM T11448 C8OZ2X 10401405 Ki = 4350 nM T11448 CR4LS0 10430623 Ki > 5000 nM T11448 CIQ02H 10436842 Ki = 4519 nM T11448 CIDE58 10473701 Ki = 895 nM T11448 C8FA2T 10474679 Ki = 1850 nM T11448 CBS8U6 10475736 Ki = 1320 nM T11448 CW81LP 10480357 Ki = 2.9 nM T11448 CJ0K1T 10507651 Ki = 954.99 nM T11448 C2U8AC 10508016 Ki = 1584.89 nM T11448 C4XZ3Y 10508132 Ki = 954.99 nM T11448 CZP09X 10508332 Ki = 630.96 nM T11448 C4X9EF 10531532 Ki = 446.68 nM T11448 C7MI2N 10531766 Ki = 1122.02 nM T11448 CF24MW 10579368 Ki = 1174.9 nM T11448 CW2HX7 10584556 Ki = 3200 nM T11448 CK8SO7 10603951 Ki = 676.08 nM T11448 C1DXO0 10609673 Ki = 130 nM T11448 CB26QH 10626982 Ki = 630.96 nM T11448 CSWC40 10627021 Ki = 1288.25 nM T11448 CF1P6Z 10651080 Ki = 501.19 nM T11448 C3K7UP 10651654 Ki = 912.01 nM T11448 CTB7L2 10674896 Ki = 758.58 nM T11448 CTSY18 10682720 Ki = 39 nM T11448 C3IX8A 10707358 Ki = 1.445 nM T11448 CT1K3B 10769331 Ki = 109.65 nM T11448 CW6GY4 10775000 Ki = 8.71 nM T11448 C3O7YN 10793665 Ki = 2137.96 nM T11448 C0D6MW 10793963 Ki = 645.65 nM T11448 CBO8N9 10818003 Ki = 676.08 nM T11448 CE80NV 10841190 Ki = 2187.76 nM T11448 CYSL64 10841387 Ki = 398 nM T11448 C0KZU8 10847653 Ki = 1.259 nM T11448 C5AY9R 10848826 Ki = 20.89 nM T11448 C4SBO9 10915140 IC50 = 3100 nM T11448 C8VT6G 10916464 Ki = 5011.87 nM T11448 CH95TI 10923927 Ki = 794.33 nM T11448 C3CI6Z 10934575 EC50 = 25.12 nM T11448 CGW87Y 11034737 Ki = 199.53 nM T11448 CA7IB5 11043720 Ki = 186.21 nM T11448 C48QYR 11058166 Ki = 870.96 nM T11448 C7JI1M 11059195 Ki < 7943.28 nM T11448 C7R2AZ 11079593 Ki = 398.11 nM T11448 C91BKL 11090351 Ki < 7943.28 nM T11448 CFE1M7 11097789 Ki = 58.88 nM T11448 CTG4I5 11098175 EC50 = 199.53 nM T11448 CR6K4V 11109088 EC50 = 6.31 nM T11448 C6SXJ0 11140033 Ki = 91.2 nM T11448 CG40BP 11140345 EC50 = 100 nM T11448 CO0XW1 11140347 Ki = 18.2 nM T11448 CTA5J4 11173544 Ki = 41.69 nM T11448 CU86DN 11173568 Ki = 37.15 nM T11448 C8V3GQ 11183468 Ki = 72.44 nM T11448 C5JYO7 11186227 Ki = 33.88 nM T11448 C0W4SM 11186523 Ki = 156 nM T11448 C1VIN4 11190988 Ki = 1.3 nM T11448 CHU5B0 11191321 Ki = 4.7 nM T11448 C3ALW8 11199581 Ki = 309.03 nM T11448 C9T7YZ 11199593 Ki = 338.84 nM T11448 C01AFD 11200476 Ki = 1.6 nM T11448 C5YQ0F 11203101 Ki = 29 nM T11448 C24JXQ 11204090 IC50 = 47 nM T11448 C62KQF 11211035 Ki = 14.79 nM T11448 CYQ65M 11214030 Ki = 0.7 nM T11448 CEGZ35 11221758 Ki = 173.78 nM T11448 CV2R8E 11224953 Ki = 20 nM T11448 C59VOU 11225732 Ki = 304 nM T11448 C3RO9W 11225779 Ki = 0.3 nM T11448 COCU26 11246610 Ki = 123.03 nM T11448 CXNM72 11259744 Ki = 0.4 nM T11448 C5PWC6 11260018 Ki = 0.9 nM T11448 CNTE30 11265631 Ki = 138.04 nM T11448 CZ8DY9 11271808 Ki = 0.1 nM T11448 C8SYW5 11277479 Ki = 51.29 nM T11448 C84NSM 11278634 Ki < 10000 nM T11448 CCWK17 11284878 IC50 = 110 nM T11448 CNAQ56 11293787 Ki = 857 nM T11448 CA1D3O 11300487 Ki = 46.77 nM T11448 C7VS0M 11306100 Ki = 0.1 nM T11448 CM67PT 11318438 Ki = 1 nM T11448 C3JBI0 11338418 Ki > 500 nM T11448 CR1K5W 11342160 IC50 = 170 nM T11448 C96OKG 11346584 Ki = 27.54 nM T11448 CGPH62 11347303 Ki = 22.91 nM T11448 CV17WA 11360447 Ki = 16.98 nM T11448 CI69GW 11361608 Ki = 60.26 nM T11448 CA28SQ 11371902 Ki = 45.71 nM T11448 C9U5WT 11380132 Ki = 1202.26 nM T11448 C1ZOY6 11380133 Ki = 281.84 nM T11448 C4JVS8 11385652 Ki = 33 nM T11448 CB01AS 11448533 Ki = 8128.31 nM T11448 CX8CN6 11473729 Ki = 8128.31 nM T11448 C1JC8F 11608298 Ki = 3600 nM T11448 CZA0M9 11653915 Ki = 6.3 nM T11448 CJ1KW9 11741010 Ki = 650 nM T11448 CPG15O 11743399 IC50 > 1000 nM T11448 CIM1E0 11750482 Ki = 204 nM T11448 CJ58LT 11765813 Ki = 0.76 nM T11448 CH8F9N 11775717 IC50 = 580400 nM T11448 CZYB79 11777109 Ki = 3 nM T11448 CX7PJ0 11779076 IC50 > 300000 nM T11448 CX7TO1 11785068 Ki = 0.9 nM T11448 CE4Q9W 11785961 Ki = 1.3 nM T11448 CFTI34 11801828 Ki = 2089.3 nM T11448 C1VWL5 11811395 Ki = 2951.21 nM T11448 CN9H3J 11820372 IC50 = 3000 nM T11448 CXLW54 11948707 Ki = 250 nM T11448 CWB20E 11957683 Ki = 1.905 nM T11448 C8JQL7 11957735 IC50 > 10000 nM T11448 CGY20U 12114850 Ki = 26.4 nM T11448 CNS58C 12114851 Ki = 15.3 nM T11448 CVY50Z 12114852 Ki = 0.87 nM T11448 C7DQR1 12114853 Ki = 1.25 nM T11448 CIUR20 12699315 Ki = 1949.84 nM T11448 C2U3RT 12764879 EC50 > 10000 nM T11448 C0B1QO 12764880 EC50 > 10000 nM T11448 CM0DW4 12981867 Ki = 39.81 nM T11448 CQ2W8P 12981869 Ki = 158.49 nM T11448 C5NPY6 12981870 Ki = 19.95 nM T11448 C2V9FL 13091268 Ki = 2835 nM T11448 CY7A4L 13869716 Ki = 42657.95 nM T11448 C7TJX3 15463615 Ki = 31.62 nM T11448 C1CX2S 15675860 Ki = 74.13 nM T11448 CXW37K 15987265 IC50 = 310 nM T11448 C0G2EO 16007117 Ki = 455 nM T11448 C1SR0O 16071847 Ki > 5000 nM T11448 CXM74T 16090594 Ki = 850 nM T11448 C8QLC1 16090595 Ki = 910 nM T11448 C01RFM 16090596 Ki = 1900 nM T11448 CAYX52 16090597 Ki = 2300 nM T11448 CW0U8R 16090598 Ki = 775 nM T11448 C06KXJ 16090599 Ki > 10000 nM T11448 COB96N 16090600 Ki = 1000 nM T11448 C6YPM3 16090601 Ki = 1870 nM T11448 CR02MW 16090602 Ki = 2200 nM T11448 CC5HV2 16090621 Ki = 580 nM T11448 COTF82 16090622 Ki = 1400 nM T11448 CB2Z6H 16090623 Ki = 790 nM T11448 C4WAZ1 16090624 Ki = 1050 nM T11448 C6MH3Z 16090625 Ki = 680 nM T11448 CX98OC 16090626 Ki = 1230 nM T11448 C6D0WK 16090627 Ki = 900 nM T11448 C1B5TL 16090628 Ki = 8000 nM T11448 CTXU32 16090630 Ki = 1170 nM T11448 CD8FX2 16090631 Ki = 3100 nM T11448 C63QEJ 16090632 Ki = 9600 nM T11448 C98XNF 16090633 Ki = 980 nM T11448 C1G7KL 16090634 Ki = 3600 nM T11448 C8YBI4 16090635 Ki = 630 nM T11448 CQS4V1 16112801 IC50 > 1000 nM T11448 CZ1WJ4 16117151 Ki > 5000 nM T11448 CM32ZX 16117153 Ki > 5000 nM T11448 CXTB90 16117279 Ki > 5000 nM T11448 C1F2LS 16118795 Ki > 5000 nM T11448 C69VDS 16118923 Ki > 5000 nM T11448 C1YWG6 16215415 Ki = 69 nM T11448 CZ2IS9 16660294 Ki > 10000 nM T11448 C3JV0P 16718827 IC50 > 1000 nM T11448 C3YN5S 16718917 IC50 = 700 nM T11448 CJ8Y1H 16718919 IC50 = 1213 nM T11448 CB7G3R 16718920 IC50 > 1000 nM T11448 CVU96E 16725934 Ki = 1742 nM T11448 CFMX86 16757089 Ki = 81.28 nM T11448 C6OJ3A 16757182 Ki = 72.44 nM T11448 CM60NI 17804479 EC50 = 722 nM T11448 C6AOE8 19426635 IC50 = 436.52 nM T11448 CPRJ25 21392988 Ki = 16595.87 nM T11448 C3T5HF 21509921 Ki = 228 nM T11448 CJD1K4 21584368 Ki = 3900 nM T11448 CT7XG9 21830793 Ki = 96 nM T11448 C8GUJ3 22120322 IC50 = 0.3467 nM T11448 CGO3B8 22120332 IC50 = 0.2951 nM T11448 C02AEX 22493245 Ki < 7943.28 nM T11448 C81XUE 23027035 IC50 = 1770 nM T11448 CR5H1I 23027211 IC50 = 130 nM T11448 CC2L1B 23027245 IC50 = 730 nM T11448 CG9M4Y 23027411 IC50 = 1590 nM T11448 CC6R2O 23027527 IC50 = 470 nM T11448 C3B0XJ 23292293 Ki = 25.12 nM T11448 CF9D1U 23622576 Ki = 74.13 nM T11448 CL4WV2 24180125 IC50 = 2830 nM T11448 CD7CV6 24771120 Ki > 2000 nM T11448 CDC91N 24839550 Ki = 123.03 nM T11448 CY21RE 24841480 Ki = 95 nM T11448 C2C7WN 24882007 Ki = 52 nM T11448 C2LV1U 24882019 EC50 = 37 nM T11448 C54TLD 24882106 EC50 = 180 nM T11448 C8WH5Z 24906160 Ki = 660.69 nM T11448 C3RQ1P 24906196 Ki = 416.87 nM T11448 CBT65R 24906197 Ki = 213.8 nM T11448 C9OAG1 24906198 Ki = 57.54 nM T11448 CYL83G 24906199 Ki = 50.12 nM T11448 CC9W0R 24906200 Ki = 239.88 nM T11448 CYEA86 24906201 Ki = 724.44 nM T11448 CIR8G1 24906202 Ki = 281.84 nM T11448 CPH75D 24906203 Ki = 398.11 nM T11448 CBUH25 24906241 Ki = 239.88 nM T11448 CUNP93 24906242 Ki = 257.04 nM T11448 C7Y2SB 24906243 Ki = 125.89 nM T11448 C1VRJ3 25014630 IC50 = 24000 nM T11448 CMVL70 25059766 IC50 > 1000 nM T11448 CED30A 25059770 IC50 > 1000 nM T11448 CJU9Y7 25060021 IC50 > 1000 nM T11448 C36PMH 25060023 IC50 > 1000 nM T11448 CHSB87 25060024 IC50 > 1000 nM T11448 CJOY17 25066019 EC50 > 10000 nM T11448 CYJ5G1 25067564 Ki > 10000 nM T11448 C9XMH7 25110718 Ki = 94.4 nM T11448 CX04LB 25142456 Ki = 180 nM T11448 CDQ70A 25208878 IC50 = 1097 nM T11448 CJ1Z9H 25216680 Ki > 3000 nM T11448 C1T3LR 25218143 Ki > 3000 nM T11448 CPI03N 25218397 Ki > 3000 nM T11448 CL1R3Q 25218401 Ki > 3000 nM T11448 CM2T9Y 25263297 Ki > 2000 nM T11448 CFJM71 25263302 Ki > 2000 nM T11448 C4MRQ0 27842480 Ki > 10000 nM T11448 CWT9F7 28918670 Ki = 95.5 nM T11448 CDP76A 42266865 Ki = 1.69 nM T11448 CP54VF 42267840 Ki = 5.19 nM T11448 CWOL80 42273326 Ki = 4.59 nM T11448 CG56DF 42388639 Ki = 4.64 nM T11448 CY7W2J 42631003 Ki = 1.995 nM T11448 CJ3NP5 42636941 IC50 = 891.25 nM T11448 CJ41QV 44126269 Ki = 0.8128 nM T11448 C2AV1K 44190762 IC50 = 1650 nM T11448 C9O1RI 44215744 Ki = 5 nM T11448 CTR42S 44219718 Ki > 2780 nM T11448 CK7F2E 44240743 IC50 = 35000 nM T11448 CL09IQ 44263496 IC50 > 10000 nM T11448 C87MXH 44263497 IC50 > 1000 nM T11448 CO65VL 44269006 Ki = 125.89 nM T11448 C0TP2Z 44269013 Ki = 48.98 nM T11448 CW6A9E 44269089 Ki = 72.44 nM T11448 CZ63DE 44269122 Ki = 26.92 nM T11448 CDS8G5 44269140 Ki = 83.18 nM T11448 CZ5P6U 44288769 Ki = 3388 nM T11448 CZ7O4D 44288847 Ki = 7852 nM T11448 C6DYQ1 44288874 Ki = 1972 nM T11448 CAG7E1 44288877 Ki = 13646 nM T11448 CQ3Y5R 44288945 Ki = 229 nM T11448 C5ZL4A 44289035 Ki = 1862 nM T11448 CLRZ30 44292232 EC50 = 10.96 nM T11448 C7GUL1 44292381 Ki = 18.2 nM T11448 C3G1KO 44292385 Ki = 13.8 nM T11448 C0R8WU 44292386 Ki = 15.85 nM T11448 C6G8ZC 44311789 Ki = 14791.08 nM T11448 C5L1WN 44312036 Ki = 3801.89 nM T11448 CT46CK 44312037 EC50 = 2754.23 nM T11448 C3XFH4 44312198 Ki = 26302.68 nM T11448 CZ4TN0 44314198 EC50 = 1.622 nM T11448 CCI07K 44314200 Ki = 25.7 nM T11448 CV8WZ0 44318454 IC50 = 501.19 nM T11448 CXJL56 44318842 IC50 > 1000 nM T11448 CA56FM 44324725 Ki = 26 nM T11448 CW16JD 44324737 Ki = 1.3 nM T11448 CA84SN 44324765 Ki = 2.6 nM T11448 COA3H4 44324800 Ki = 0.3 nM T11448 CK32IL 44324859 Ki = 22 nM T11448 CMB1S6 44324860 Ki = 98 nM T11448 C8HUD2 44324887 Ki = 0.8 nM T11448 CCT53K 44324900 Ki = 186 nM T11448 CL1F3T 44324906 Ki = 0.5 nM T11448 CPAL75 44324937 Ki = 0.9 nM T11448 CY04JW 44324972 Ki = 0.3 nM T11448 C76UJT 44325027 Ki = 34 nM T11448 C1RS8C 44325028 Ki = 234 nM T11448 CR4Q1C 44325038 Ki = 117 nM T11448 C4SZJ2 44325044 Ki = 66 nM T11448 CQX1Y0 44325049 Ki = 1.4 nM T11448 C0N3JG 44325050 Ki = 0.8 nM T11448 CEYD96 44325075 Ki = 12 nM T11448 CGS4E7 44325079 Ki = 234 nM T11448 CV7L8H 44330114 Ki = 0.5 nM T11448 C7Q1HP 44330168 Ki = 0.3 nM T11448 COY19U 44330368 Ki = 1.9 nM T11448 C1Z6DB 44330369 Ki = 1.4 nM T11448 CKO67I 44330427 Ki = 3 nM T11448 CP7Y9I 44330571 Ki = 23 nM T11448 C3AY4O 44330584 Ki = 2.9 nM T11448 CVTA63 44330598 Ki = 5.9 nM T11448 C83NZA 44330609 Ki = 9 nM T11448 C2AOH6 44330617 Ki = 1.1 nM T11448 C2RQ3Z 44330621 Ki = 69 nM T11448 C7JP2X 44330635 Ki = 1 nM T11448 CCVE83 44330645 Ki = 1.7 nM T11448 CO8XC7 44330653 Ki = 1.7 nM T11448 C47ZPQ 44330668 Ki = 1.1 nM T11448 CGJ05Y 44330679 Ki = 22 nM T11448 C9D2SN 44330857 Ki = 5.2 nM T11448 C6N3XK 44345317 IC50 < 1000 nM T11448 CZ2X3A 44352155 EC50 = 63.1 nM T11448 C67ZNM 44352207 Ki = 47.86 nM T11448 C6KJV8 44371744 Ki = 16.6 nM T11448 CI90WF 44371745 Ki = 23.99 nM T11448 C09ADW 44371755 Ki = 11.75 nM T11448 CUF64I 44371848 Ki = 1.18 nM T11448 C76VTG 44371864 EC50 = 11.75 nM T11448 C3K6GE 44376845 IC50 = 3.548 nM T11448 CPD18R 44376900 IC50 = 0.6918 nM T11448 CE46SW 44376923 IC50 = 0.2884 nM T11448 C7UW8Z 44376927 IC50 = 1.175 nM T11448 C8GT5O 44376936 IC50 = 10.23 nM T11448 CLC2T4 44376954 IC50 = 0.3388 nM T11448 C9IPC3 44376958 IC50 = 0.4467 nM T11448 CX4A1Z 44376975 IC50 = 2.188 nM T11448 C14SMK 44376984 IC50 = 0.2399 nM T11448 C0V4XL 44376993 IC50 = 0.5888 nM T11448 CX0UR3 44377006 IC50 = 3.89 nM T11448 CB2R0M 44377007 IC50 = 0.8913 nM T11448 C2ID6U 44377035 IC50 = 0.6026 nM T11448 C6R9OZ 44377036 IC50 = 0.2138 nM T11448 C97QIG 44377200 IC50 = 0.3548 nM T11448 C93JCM 44387789 Ki = 0.5 nM T11448 CI52GK 44387798 Ki = 47 nM T11448 CE25YT 44390369 IC50 = 34 nM T11448 CFH3C2 44390385 IC50 = 31 nM T11448 C6LJC2 44390456 IC50 = 44 nM T11448 CHGY52 44390499 IC50 = 9.9 nM T11448 CK7G4S 44390706 IC50 = 63 nM T11448 CS16BQ 44390710 IC50 = 60 nM T11448 C9GTA2 44390713 IC50 = 130 nM T11448 C0B5MU 44390715 IC50 = 47 nM T11448 CBA36Y 44390726 IC50 = 71 nM T11448 C9GTB7 44390730 IC50 = 150 nM T11448 CPQ63J 44390733 IC50 = 170 nM T11448 CHO04I 44390742 IC50 = 150 nM T11448 CZN1R2 44390750 IC50 = 76 nM T11448 C3TEB2 44390752 IC50 = 520 nM T11448 C85MAY 44390768 IC50 = 97 nM T11448 C5BA0Y 44390778 IC50 = 110 nM T11448 CN3U4V 44390787 IC50 = 200 nM T11448 CX7O9S 44401041 Ki = 269 nM T11448 C5XC2B 44401042 Ki = 302 nM T11448 CD56EA 44401105 Ki = 407 nM T11448 CW3PC2 44401106 Ki = 72 nM T11448 C9WH7P 44401164 Ki = 66 nM T11448 C9CWX1 44401194 Ki = 251 nM T11448 CXT84G 44401243 Ki = 10 nM T11448 C4RN8A 44401449 IC50 = 57 nM T11448 C49USD 44401460 IC50 = 86 nM T11448 CHGX51 44401508 IC50 = 58 nM T11448 CIKD90 44401552 IC50 = 140 nM T11448 C8VQ3B 44401591 IC50 = 100 nM T11448 CT46VH 44401616 IC50 = 21 nM T11448 CIXE76 44401626 IC50 = 130 nM T11448 CER15G 44401671 IC50 = 5.6 nM T11448 C6YP8T 44404321 Ki = 4.16 nM T11448 CYA37J 44404326 Ki = 4.73 nM T11448 CU2FG6 44415569 Ki = 169 nM T11448 CDU6Y5 44415593 Ki = 882 nM T11448 CH0BY5 44415672 Ki = 2000 nM T11448 CK59CO 44415689 Ki = 327 nM T11448 C7AZ5D 44415690 Ki = 791 nM T11448 CEVY54 44415704 Ki = 456 nM T11448 CI47TG 44421258 Ki = 1230.27 nM T11448 CK7HF3 44424855 Ki = 9 nM T11448 C28OZL 44438147 Ki = 400 nM T11448 CKB9O7 44438148 Ki = 135 nM T11448 C1AR8P 44438152 Ki = 2552 nM T11448 CZR64Y 44438161 Ki = 216 nM T11448 CG38YN 44438165 Ki = 454 nM T11448 C8RC7O 44438166 Ki = 141 nM T11448 C5GPZ7 44438167 Ki = 42 nM T11448 C0QI8L 44438168 Ki = 186 nM T11448 C64POV 44449245 EC50 > 10000 nM T11448 CX7Z6I 44449247 EC50 = 327 nM T11448 CN9BI4 44449276 EC50 = 4340 nM T11448 CYM30S 44449277 EC50 = 27 nM T11448 CS5WB3 44449278 EC50 > 10000 nM T11448 CH74NV 44449303 EC50 > 10000 nM T11448 C8VO6A 44449304 EC50 > 10000 nM T11448 CI4T2K 44449305 EC50 > 10000 nM T11448 C0M7UN 44449337 EC50 > 10000 nM T11448 C1O6QI 44449657 EC50 > 10000 nM T11448 C6QCN8 44449686 EC50 > 10000 nM T11448 CH5RL7 44449690 EC50 > 10000 nM T11448 CS3LB0 44449691 EC50 = 4580 nM T11448 CFL25O 44449692 EC50 > 10000 nM T11448 CSZB25 44449694 EC50 > 10000 nM T11448 CJ8WL7 44449723 EC50 > 10000 nM T11448 C8XHB5 44449724 EC50 > 10000 nM T11448 C6ZG3O 44449725 EC50 > 10000 nM T11448 CMLE59 44449730 EC50 > 10000 nM T11448 CZL97F 44455426 Ki > 10000 nM T11448 C12XGE 44456400 Ki = 283 nM T11448 CQ2IX7 44461606 IC50 > 1000 nM T11448 C3D4HR 44537940 Ki > 5000 nM T11448 C4LUK7 44549156 Ki = 22.91 nM T11448 CJ7U3K 44554227 Ki > 5000 nM T11448 CM0I1P 44554393 Ki > 5000 nM T11448 CNHA47 44554395 Ki > 5000 nM T11448 C8N3ID 44568614 Ki = 93.33 nM T11448 CVF30Y 44574044 Ki > 4500 nM T11448 CCD72N 44574045 Ki = 213 nM T11448 CMS20J 44574074 Ki > 3800 nM T11448 C92YUA 44574075 Ki = 805 nM T11448 C9NU2C 44574076 Ki = 1020 nM T11448 CB8US6 44574077 Ki = 1750 nM T11448 CX4Y0K 44574078 Ki = 991 nM T11448 CU9X8G 44574079 Ki = 112 nM T11448 C62FCK 44574080 Ki = 380 nM T11448 CAT57X 44574103 Ki = 1100 nM T11448 CXZ0J3 44574104 Ki = 114 nM T11448 CES4X0 44574105 Ki = 280 nM T11448 C62AYR 44574106 Ki = 202 nM T11448 CX98MY 44574107 Ki > 2370 nM T11448 CDER54 44574132 Ki > 3310 nM T11448 C4S2OQ 44574133 Ki > 2160 nM T11448 C96NQZ 44574134 Ki = 469 nM T11448 CKR69S 44574135 Ki = 1470 nM T11448 CG0RM2 44574138 Ki > 3230 nM T11448 CD87ZE 44574834 EC50 > 10000 nM T11448 CWM4U7 44579184 Ki = 167 nM T11448 CLO8A9 44579185 Ki = 220 nM T11448 CGVM03 44579186 Ki = 27 nM T11448 CM6L2Y 44579187 Ki = 208 nM T11448 CBDL39 44579228 Ki = 138 nM T11448 CX5O1H 44579229 Ki = 73.6 nM T11448 C3G5YK 44579230 Ki = 48.4 nM T11448 CKTJ23 44579231 Ki = 443 nM T11448 C57BWM 44579271 Ki = 66.1 nM T11448 C7R9XM 44579272 Ki = 15.4 nM T11448 CRCH48 44582675 Ki > 10000 nM T11448 CEJ4R8 44582676 Ki = 863 nM T11448 C5QB4K 44582678 Ki > 10000 nM T11448 C9F6EB 44593557 Ki > 1700 nM T11448 C51AJZ 44593577 EC50 > 10000 nM T11448 CF3T8K 44596863 IC50 = 320 nM T11448 CWO70X 45260703 Ki = 977.24 nM T11448 C4VOW6 45260704 Ki = 81.28 nM T11448 CQ0R5Y 45264581 EC50 = 39.81 nM T11448 C39CDN 45264638 Ki = 81.28 nM T11448 C0CHF4 45482789 IC50 = 1930 nM T11448 CGLF37 45484995 IC50 = 210 nM T11448 CGOS24 45485061 IC50 = 200 nM T11448 CLX9C8 45485062 IC50 = 580 nM T11448 CQHW85 45487089 Ki = 24.55 nM T11448 CI34PT 45487144 Ki = 26.92 nM T11448 CC9GH0 45487145 Ki = 57.54 nM T11448 C7MZ9Y 45487955 Ki = 50.12 nM T11448 CLW5M9 45487956 Ki = 22.91 nM T11448 C45DAV 45487958 Ki = 34.67 nM T11448 CZSW97 45487962 Ki = 48.98 nM T11448 C5FQ4S 46224879 Ki = 0.2399 nM T11448 CY82LR 46227396 IC50 = 891 nM T11448 C03LTM 46869265 Ki = 3500 nM T11448 CK8A1O 46880462 Ki > 10000 nM T11448 C9KDP4 46880463 Ki > 10000 nM T11448 CODR73 46880498 Ki > 10000 nM T11448 CHJ5Y6 46880566 Ki > 10000 nM T11448 CE9PG2 46880567 Ki > 10000 nM T11448 C01PGO 46880568 Ki > 10000 nM T11448 CS7L4X 46880569 Ki > 10000 nM T11448 C0PXY7 46880628 Ki > 10000 nM T11448 CD37LU 46880629 Ki > 10000 nM T11448 CUY89F 46880630 Ki > 10000 nM T11448 C4P6XS 46880631 Ki > 10000 nM T11448 CJ53KF 46880672 Ki > 10000 nM T11448 CYJC08 46880673 Ki > 10000 nM T11448 C1RI9O 46880674 Ki > 10000 nM T11448 CJ6K2R 46891598 Ki = 1.6 nM T11448 CZDN92 46934426 Ki = 11.1 nM T11448 C4VG2E 46934427 Ki = 2.87 nM T11448 C8VUO2 49781004 Ki = 11.75 nM T11448 C0LAT9 49781005 Ki = 0.5623 nM T11448 C12UVE 49781006 Ki = 3.311 nM T11448 CW1V4K 49781007 Ki = 3.981 nM T11448 CF9L7Z 49781008 Ki = 45.71 nM T11448 CQ2EN5 49781222 Ki = 0.2188 nM T11448 CV62OU 49781223 Ki = 0.5129 nM T11448 C3I5HP 49781224 Ki = 0.8511 nM T11448 CF5CO4 49781228 Ki = 0.02818 nM T11448 CW5X6A 49781887 Ki = 0.3311 nM T11448 C2LZJ0 49783209 Ki = 2239 nM T11448 C57SMG 49783415 Ki > 10000 nM T11448 C0TG6I 49783419 Ki > 10000 nM T11448 C28CKM 49836301 Ki = 52.48 nM T11448 C5JO6E 49836302 Ki = 100 nM T11448 C9TNO4 49836303 Ki = 20.89 nM T11448 CL6QA1 49836304 Ki = 44.67 nM T11448 CE1S9B 49836305 Ki = 44.67 nM T11448 CP0DJ4 49836306 Ki = 165.96 nM T11448 CJM3F9 49836307 Ki = 97.72 nM T11448 C0LN3I 49836308 Ki = 39.81 nM T11448 C8TB6G 49864336 Ki = 4.1 nM T11448 C5N8ML 49864359 Ki = 8.53 nM T11448 C15NIO 49864360 Ki = 6.15 nM T11448 C2RY0J 50878551 Ki = 213.8 nM T11448 C1W6TV 50898777 Ki > 10000 nM T11448 CXMZ73 50898778 Ki > 10000 nM T11448 CS2Z6C 50994258 EC50 = 14 nM T11448 CS24VY 50994260 EC50 = 73 nM T11448 CE4KP1 51050257 Ki > 10000 nM T11448 CR8MI3 52941512 Ki = 0.1738 nM T11448 CZ4SA1 52942940 Ki = 1513.56 nM T11448 CH3YE5 52943739 Ki = 0.4467 nM T11448 C70LBS 52944548 Ki = 0.138 nM T11448 C7WN4S 52948958 Ki = 0.4074 nM T11448 C5W7SH 52950140 Ki = 1.072 nM T11448 C12VMW 53322686 EC50 = 82 nM T11448 C4IPV8 53323136 EC50 = 15 nM T11448 C8KRS1 53324490 EC50 = 240 nM T11448 CR4W9L 53324553 Ki = 7609 nM T11448 C2KG9D 56665110 Ki > 10000 nM T11448 C5E1XF 56729561 Ki = 141.25 nM T11448 CJKO58 56852956 Ki = 844 nM T11448 CL16UQ 56949326 IC50 < 10000 nM T11448 C5O2XV 56950526 EC50 = 16600 nM T11448 C1TC7Q 56963799 Ki > 10000 nM T11448 CUL4N1 56964693 Ki = 729 nM T11448 CQ5TP0 56964794 Ki = 374 nM T11448 C20ILW 57326584 Ki = 412 nM T11448 C1ZO5L 57326586 Ki = 452 nM T11448 CL45WN 57345320 IC50 = 3700 nM T11448 C4RBY6 57345625 Ki = 28.84 nM T11448 C1US6F 57345626 Ki = 22.91 nM T11448 CNU83J 57345627 Ki = 72.44 nM T11448 CD50GK 57345628 Ki = 36.31 nM T11448 C4FA1T 57345629 Ki = 83.18 nM T11448 CO2W7Z 57384051 Ki = 398.11 nM T11448 C3M7AS 57391904 EC50 = 4500 nM T11448 C80DHR 57393066 Ki > 10000 nM T11448 C6X0ZI 57394788 Ki = 5370.32 nM T11448 CR6U3P 57394789 Ki = 6309.57 nM T11448 CH84EC 57395663 Ki = 181.97 nM T11448 CL37YV 57395731 EC50 = 63.1 nM T11448 C5I3DG 57395732 Ki = 489.78 nM T11448 CR1Y7M 57398332 Ki = 501.19 nM T11448 CM9WK5 57399145 Ki = 97.72 nM T11448 CIB2L3 57399991 Ki = 7943.28 nM T11448 C1CW6M 57400570 EC50 = 17400 nM T11448 CQ7MC1 57400959 EC50 = 562.34 nM T11448 C9WE2A 57401787 Ki = 3801.89 nM T11448 C56WAY 57402717 Ki = 57.54 nM T11448 C1BFP4 57402718 EC50 = 31.62 nM T11448 CP21KC 57403508 Ki > 10000 nM T11448 C2PJ4N 59271992 IC50 = 1000 nM T11448 CD3U6K 68731121 Ki > 3000 nM T11448 C6IP8Q 69082816 Ki > 3000 nM T11448 CLM79R 70686398 Ki > 10000 nM T11448 CJQX48 70693375 Ki = 44.67 nM T11448 CST13M 70695474 Ki = 41.69 nM T11448 C6CNI0 70696790 Ki = 4897.79 nM T11448 CKD60A 70789640 Ki = 1416 nM T11448 C9VZ8J 71450550 Ki = 1301 nM T11448 CGQ0R2 71450907 Ki = 0.9 nM T11448 CTDN12 71452341 Ki = 1232 nM T11448 CE0R9D 71454275 Ki = 17170 nM T11448 CUX98O 71456238 Ki = 11 nM T11448 COG3Y0 71456239 Ki = 43 nM T11448 CYR3D4 71456240 Ki = 1.8 nM T11448 C5DLQ2 71459553 Ki = 653 nM T11448 CR3LH2 71461647 Ki = 1.8 nM T11448 CL91AC 71463022 Ki = 945 nM T11448 C3ATN5 72197484 IC50 > 10000 nM T11448 CN8A5R 72197486 IC50 > 10000 nM T11448 C5L8NJ 72947314 Ki = 77.62 nM T11448 CE1JY2 72947315 Ki = 316.23 nM T11448 CC65OA 73213195 Ki = 1800 nM T11448 CW83DK 73213196 Ki = 407 nM T11448 C02FTM 73291731 Ki = 50.12 nM T11448 CCV91B 73346042 Ki = 2751 nM T11448 CK0HR9 73346334 Ki > 10000 nM T11448 C6J0TM 73346336 Ki > 10000 nM T11448 CR97NO 73347825 Ki = 5211 nM T11448 CH2B4Y 73350932 Ki > 10000 nM T11448 C2E7QW 75201901 Ki = 3400 nM T11448 C8IDL3 75306277 Ki = 63.1 nM T11448 CBRI02 78114597 Ki = 0.3236 nM T11448 CMF3A7 78114671 Ki = 9549.93 nM T11448 C8JFM6 78114674 Ki = 0.0537 nM T11448 CR6Z8F 78114676 Ki = 3.236 nM T11448 CTS2P9 78114881 Ki = 4.467 nM T11448 C5YCX6 90644701 Ki = 1479.11 nM T11448 CNHV06 90644703 Ki = 213.8 nM T11448 CIKB60 90644705 Ki = 512.86 nM T11448 CK46DZ 90644707 Ki = 1071.52 nM T11448 C6GZC4 90644709 Ki = 1513.56 nM T11448 CT86PS 90644711 Ki = 19054.61 nM T11448 COLI89 90644713 Ki = 1862.09 nM T11448 C8KXV4 90644715 Ki = 1737.8 nM T11448 C0N1HX 90644717 Ki = 18620.87 nM T11448 C50DUP 90644719 Ki = 11748.98 nM T11448 CU5I3L 90644721 Ki = 2238.72 nM T11448 CTP9A6 90644723 Ki = 389.05 nM T11448 CE7MA4 90644725 Ki = 3311.31 nM T11448 CLK04X 90644727 Ki = 1000 nM T11448 CM2I8Y 90644729 Ki = 12302.69 nM T11448 CH2CE6 90644731 Ki = 2344.23 nM T11448 CT7SG6 90644733 Ki = 2630.27 nM T11448 C47LDA 90644735 Ki = 1318.26 nM T11448 C12XVI 90644737 Ki = 691.83 nM T11448 C45ASR 90644739 Ki = 2187.76 nM T11448 C1V0IO 90644741 Ki = 1698.24 nM T11448 CX6LE2 90644743 Ki = 79.43 nM T11448 C7PZO5 90644745 Ki = 263.03 nM T11448 CTER62 90644747 Ki = 4897.79 nM T11448 CSW20Z 90644749 Ki = 4365.16 nM T11448 C0U8RJ 90644750 Ki = 4265.8 nM T11448 C2Q5PD 90644751 Ki = 1122.02 nM T11448 CJZX10 90644752 Ki = 676.08 nM T11448 C8LZ9W 90644754 Ki = 8317.64 nM T11448 C5A8WP 90644756 Ki = 15135.61 nM T11448 C1G3ZC 90644757 Ki = 14125.38 nM T11448 CUQ6V0 92042918 Ki < 1000 nM T11448 CGC29J 92042920 Ki < 1000 nM T11448 C7YQM3 101333429 Ki = 1550 nM T11448 C90GPJ 103616908 Ki = 11000 nM T11448 CWR6I1 118112300 IC50 = 8000 nM T11448 CUV5Y0 118715454 EC50 > 30000 nM T11448 CCY5S0 118717248 Ki = 33 nM T11448 CCR09Q 118717249 Ki = 65 nM T11448 C5X8MN 122186880 Ki = 719 nM T11448 C7ODW3 122195524 Ki < 300 nM T11448 CM57GR 126720252 Ki = 28 nM T11448 CTBN56 127026052 Ki = 117.49 nM T11448 C8MC1I 127028408 Ki = 165.96 nM T11448 CZ61LK 127034966 IC50 > 5011.87 nM T11448 CA0SN5 127034967 EC50 > 5011.87 nM T11448 CQ0ZT9 127035062 Ki = 102 nM T11448 CU49VE 127036186 Ki = 194.98 nM T11448 CG06BD 127036932 Ki = 81.28 nM T11448 CVW71O 127036953 Ki = 83.18 nM T11448 CYJ9R5 127048642 Ki = 58000 nM T11448 C85KDT 127048643 Ki = 62000 nM T11448 C2BAM1 127048644 Ki = 80000 nM T11448 CQ8UR0 127048645 Ki = 52000 nM T11448 CZF3T9 127048646 Ki = 27000 nM T11448 CPRD68 127050218 Ki = 110000 nM T11448 C05IVG 127050224 Ki = 41000 nM T11448 C3DC8Y 127051133 Ki = 99000 nM T11448 CN05YW 127052992 Ki = 110000 nM T11448 CR8HP6 129281194 IC50 = 900 nM T11448 C50GOC 130442480 Ki = 6800 nM T11448 CM04RF 130442572 Ki = 5100 nM T11448 C1RI8Q 132060720 Ki = 1685 nM T11448 C0DIF5 132060733 Ki = 2089 nM T11448 CY8B9L 132060743 Ki = 487 nM T11448 C7FM0U 132060763 Ki = 876 nM T11448 CT81OY 132060776 Ki = 506 nM T11448 C7CSU4 132075278 Ki = 321 nM T11448 CAVB41 132584404 Ki = 1586 nM T11448 CBU81N 134149168 Ki > 10000 nM T11448 C1GY2T 135156251 EC50 > 10000 nM T11448 C2PT4I 135356876 Ki = 1560 nM T11448 CKO6D5 135405894 Ki = 9.1 nM T11448 CP58JO 135418497 Ki = 444 nM T11448 C1DFG8 135433755 Ki = 3.162 nM T11448 C7HYA8 135440165 Ki = 2.4 nM T11448 CMK06P 135477797 Ki = 6.5 nM T11448 C1IKQ6 135499867 Ki = 20 nM T11448 CTP2R6 135519400 Ki = 0.2 nM T11448 CA39PK 135519421 Ki > 1000 nM T11448 CCBM21 135545454 Ki = 7.9 nM T11448 CH96LU 135559170 Ki = 547 nM T11448 C5J9BC 136019934 Ki = 1.3 nM T11448 CXA5Y9 136044137 Ki = 74 nM T11448 CUC40S 136078488 Ki = 63.1 nM T11448 C0TAI6 136274356 Ki > 1000 nM T11448 CF7S1X 136274357 Ki = 4 nM T11448 CE8N4S 137641762 Ki = 5000 nM T11448 CKS5V0 137643541 Ki = 5000 nM T11448 CPI68E 137646281 Ki = 221 nM T11448 CLT73G 137647199 Ki = 2570 nM T11448 CI14LP 145949343 IC50 = 5900 nM T11448 CGW92C 145952721 IC50 > 30000 nM T11448 CT5CX0 145973771 Ki = 5280 nM T11448 C4GV8Q 145990586 Ki = 1147 nM T11448 CC2G1V 146025727 Ki = 2600 nM T11448 CV9G7Z 153287572 Ki > 10000 nM T11448 CO85KL 153287574 Ki = 398.11 nM T11448 CAS3E0 155510985 Ki = 169824.37 nM T11448 C75CEX 155513073 Ki = 7.762 nM T11448 CVU8Q3 155513359 Ki = 0.06607 nM T11448 CUM2N4 155515982 Ki = 400 nM T11448 C8QG2E 155517797 Ki = 48977.88 nM T11448 CTV3M6 155521287 Ki = 53 nM T11448 CT23LB 155523897 Ki = 169.82 nM T11448 CEL2K8 155525779 Ki = 602.56 nM T11448 CK8U7X 155526524 Ki = 1174.9 nM T11448 CVQ20K 155526672 Ki = 6918.31 nM T11448 CTW38M 155531234 Ki = 416869.38 nM T11448 CD5Y1E 155533747 Ki = 114815.36 nM T11448 COT9U8 155535203 Ki = 6960 nM T11448 CB79ZW 155536080 Ki = 6309.57 nM T11448 CAOH15 155538007 Ki = 4570.88 nM T11448 C7OX9U 155538461 Ki = 18620.87 nM T11448 C9S2IA 155539605 Ki = 3364 nM T11448 C08RIO 155540329 Ki = 0.04169 nM T11448 C6PE5Q 155544935 Ki = 707.95 nM T11448 C1RX8C 155545196 Ki > 1000000 nM T11448 CA7I6L 155546560 Ki > 1000000 nM T11448 CR3T5H 155546767 Ki = 25703.96 nM T11448 C02UVE 155547141 Ki = 3715.35 nM T11448 C7V2KX 155547631 Ki = 0.9772 nM T11448 CCP6V1 155550341 Ki = 63.1 nM T11448 CI06XC 155551657 Ki > 1000000 nM T11448 CX8JA1 155552185 Ki = 860 nM T11448 C3JU8M 155555790 Ki = 363078.05 nM T11448 CU0CK2 155556443 Ki = 169.82 nM T11448 CBS89O 155556618 Ki = 6800 nM T11448 C4KA3L 155566387 Ki = 141253.75 nM T11448 CYT7O8 155566429 Ki = 1412.54 nM T11448 CD1O9B 155566702 Ki = 2238.72 nM T11448 C2EO4B 155567867 Ki = 7585.78 nM T11448 CP9TR0 10324985 Ki = 1012 nM T11448 D00GEE 92766 Ki = 1218 nM T11448 D01KAX 135453290 Ki = 2270 nM T11448 D01SRL 6424833 Ki = 3200 nM T11448 D01SRS 15407445 Ki = 4840 nM T11448 D02YSX 197033 Ki = 109.65 nM T11448 D03DMN 1268096 Ki = 106 nM T11448 D03LDH 10758200 Ki = 146.1 nM T11448 D04TWX 9794475 Ki > 1000 nM T11448 D05GDP 599482 Ki = 1370 nM T11448 D05ZUX 44207909 Ki >= 1000 nM T11448 D06HHJ 10490084 Ki = 210 nM T11448 D06QKW 2765 Ki = 58.88 nM T11448 D06UBB 123981 Ki = 9.4 nM T11448 D07ICV 3072540 Ki = 3600 nM T11448 D07OAF 4038180 Ki = 33.11 nM T11448 D07QCC 10946567 Ki = 31 nM T11448 D08DOG 25130235 Ki = 74 nM T11448 D08JUO 24898732 Ki = 2238721.14 nM T11448 D08KLH 108094 Ki = 0.3631 nM T11448 D09ALJ 5280805 Ki = 9340 nM T11448 D09BIV 6455104 Ki = 46773.51 nM T11448 D09HJL 10331436 IC50 = 19000 nM T11448 D09PIN 3378093 Ki > 1000 nM T11448 D09RPR 16737207 Ki > 10000 nM T11448 D0A6GK 10489502 Ki = 95 nM T11448 D0C9DC 123920 Ki = 6520 nM T11448 D0D8GV 9830741 Ki > 45 nM T11448 D0E3OL 4567175 Ki = 720 nM T11448 D0EO4F 9891167 Ki = 82.5 nM T11448 D0F0IA 11301655 Ki > 2000 nM T11448 D0FF6S 16038374 IC50 > 10000 nM T11448 D0FU5E 10220053 Ki = 5.9 nM T11448 D0H1WR 5226 Ki = 3400 nM T11448 D0H3CW 9839317 Ki = 54 nM T11448 D0H3NA 10176567 Ki = 277 nM T11448 D0I3XA 6422124 Ki = 42.66 nM T11448 D0K0KR 9895867 IC50 = 7.7 nM T11448 D0L5MW 181743 Ki = 1288 nM T11448 D0L6JS 9816048 Ki = 9.6 nM T11448 D0L7IZ 540335 Ki = 3200 nM T11448 D0LI3J 3080926 Ki = 229.09 nM T11448 D0M5ZE 5311416 Ki = 100 nM T11448 D0M9IC 441082 Ki = 660.69 nM T11448 D0N7UE 10198248 Ki = 309.03 nM T11448 D0P5PW 132111 IC50 = 1300 nM T11448 D0PN9R 16655023 Ki = 3.1 nM T11448 D0Q7ZR 9890547 Ki = 77.8 nM T11448 D0S4VR 10655607 Ki = 76 nM T11448 D0T2RY 9948320 Ki = 530 nM T11448 D0V6DJ 5640 Ki = 612 nM T11448 D0Y0SA 135399666 EC50 = 1990 nM T11448 D0Z7EA 643606 Ki = 4.6 nM T11448 D0ZC4S 10632290 Ki = 3100 nM T01281 D0E3TC 44259 IC50 = 131 nM T01281 C3VRO9 44557921 IC50 > 10000 nM T01281 CV63UL 67240318 IC50 > 5000 nM T01281 C2MD1Q 155513187 IC50 > 10000 nM T95682 CG3PR6 52912222 IC50 > 31622.78 nM T95682 C1KWY4 54759170 IC50 = 1500 nM T95682 CM90YZ 70680608 IC50 = 4100 nM T95682 CDY89S 70680609 IC50 = 550 nM T95682 CIPN50 71760902 IC50 = 10000 nM T95682 C5TB9S 77843982 IC50 > 10000 nM T95682 COZ8S1 78319129 IC50 = 10000 nM T95682 C8BMH6 118733097 IC50 = 4000 nM T95682 CTD04M 118733098 IC50 > 50000 nM T95682 CUF52T 118733099 IC50 = 7800 nM T95682 CQ7ZG2 118733100 IC50 > 50000 nM T95682 C3Y2KO 118733101 IC50 > 50000 nM T95682 CYTV76 118733102 IC50 > 50000 nM T95682 C8A2IN 118733103 IC50 = 1010 nM T95682 C2BO5U 118733104 IC50 = 450 nM T95682 C7Q0IC 118733105 IC50 = 1380 nM T95682 CUWX94 119081692 IC50 = 880 nM T95682 C7VJH3 122512239 IC50 = 63095.73 nM T95682 C15SUJ 127025079 IC50 = 1800 nM T95682 CMG7C1 127026579 IC50 = 1800 nM T95682 CAV92O 127026580 IC50 = 1200 nM T95682 C9WLR6 127026581 IC50 = 1100 nM T95682 C57IHP 127026582 IC50 = 720 nM T95682 CM97ZL 127026583 IC50 = 1000 nM T95682 C7WE5X 127026588 IC50 = 1200 nM T95682 CB2CX8 127026589 IC50 = 1700 nM T95682 CRFG40 127026590 IC50 = 4100 nM T95682 CF9QV5 127026591 IC50 = 580 nM T95682 C6GR7I 127026628 IC50 > 30000 nM T95682 CY7T5G 127026629 IC50 = 7200 nM T95682 C3LM6B 127026630 IC50 = 3300 nM T95682 C35AYZ 127027784 IC50 = 890 nM T95682 CXL45V 127028085 IC50 = 1400 nM T95682 C0C1HZ 127028091 IC50 = 160 nM T95682 CAH3Q7 127029580 IC50 = 8600 nM T95682 CQT3A9 137636309 IC50 > 100000 nM T95682 C6YPL1 142740580 IC50 = 25118.86 nM T95682 CWE84Z 142740586 IC50 > 100000 nM T95682 CWHP86 142740595 IC50 = 316.23 nM T95682 CRK6E2 155526401 IC50 = 6309.57 nM T95682 CJ3XQ0 155531658 IC50 = 501.19 nM T95682 C02DSM 155537630 IC50 = 39810.72 nM T95682 C1TLD7 155553647 IC50 = 39810.72 nM T95682 C0JQF4 155562547 IC50 = 50118.72 nM T95682 CC8O2L 155565265 IC50 = 63095.73 nM T95682 D02KSN 91827353 IC50 = 600 nM T95682 D07HET 50967109 IC50 = 51000 nM T95682 D0I4FP 91654625 IC50 = 130 nM T95682 D0T3WL 73010930 IC50 = 400 nM T38087 D01SHZ 9931954 IC50 = 14 nM T38087 D04AIT 5280445 IC50 = 1071.52 nM T38087 D0J9HW 23725625 IC50 = 1700 nM T38087 D0Z3EI 6038 IC50 > 20000 nM T38087 D00BMF 24958200 IC50 = 5130 nM T38087 D0F5TD 135565981 IC50 = 120 nM T38087 CH62DB 1853 IC50 = 13.8 nM T38087 C5JLH9 69088 IC50 = 12000 nM T38087 CXG7Y0 76959 IC50 > 100000 nM T38087 CS74HZ 145726 IC50 = 177.83 nM T38087 C0F1IA 229015 IC50 = 310 nM T38087 CJ2UB5 236501 IC50 > 100000 nM T38087 CY65EM 261391 IC50 = 1096.48 nM T38087 CEOJ76 270800 IC50 = 5495.41 nM T38087 C7OGS2 300570 IC50 = 31200 nM T38087 CY86AM 300572 IC50 = 7244.36 nM T38087 CU2TY0 484118 IC50 = 990 nM T38087 CYC75Z 622510 IC50 = 140 nM T38087 CV7W5J 1007747 IC50 > 19000 nM T38087 C3LSW0 2088634 IC50 > 19000 nM T38087 C9R6CT 2215194 IC50 > 19000 nM T38087 C89WXS 2802462 IC50 = 72 nM T38087 C1RPD4 2807156 IC50 = 416.87 nM T38087 CJ9RE8 2818760 IC50 = 2691.53 nM T38087 CZF6C4 2867551 IC50 = 575.44 nM T38087 C1NOK3 2946601 IC50 = 1995.26 nM T38087 CZ8H1N 2959509 IC50 = 1700 nM T38087 CMX1S8 2976605 IC50 = 861 nM T38087 CAI3D8 3117362 IC50 = 15000 nM T38087 CR26SK 4163640 IC50 = 230 nM T38087 CT9V6M 4826644 IC50 = 150 nM T38087 C4C8BV 5320693 IC50 = 450 nM T38087 CB86MY 5391140 IC50 = 620 nM T38087 C7CIL3 6490174 IC50 > 100000 nM T38087 C4P2UQ 8607850 IC50 > 100000 nM T38087 CAV3P4 9899130 IC50 = 24 nM T38087 CI0QP9 11960529 IC50 = 23988.33 nM T38087 C4Y5DW 12402280 IC50 = 180 nM T38087 CQ98DR 12903736 IC50 = 11481.54 nM T38087 C0X1UV 12903737 IC50 = 354.81 nM T38087 CZ0KO4 14668434 IC50 = 36 nM T38087 CCBV16 16013151 IC50 = 509 nM T38087 CG5A7W 16013152 IC50 = 650 nM T38087 CPG4V1 16013160 IC50 = 175 nM T38087 C5ZI4W 16013163 IC50 = 1420 nM T38087 CEF0U9 16013167 IC50 = 783 nM T38087 CIA6K4 16013171 IC50 = 1100 nM T38087 CK5GZ9 16013173 IC50 = 132 nM T38087 C5IN0B 16013175 IC50 = 589 nM T38087 CK26VL 16013177 IC50 = 629 nM T38087 CW3K5S 16013181 IC50 = 2040 nM T38087 CO31UP 16013183 IC50 = 2630 nM T38087 CBMF65 16013184 IC50 = 33 nM T38087 C6V4TG 16013186 IC50 = 42 nM T38087 CZD28Q 16013188 IC50 = 1070 nM T38087 C4MIJ5 16013196 IC50 = 281 nM T38087 CJV05Q 16013198 IC50 = 197 nM T38087 C1UY7I 16013247 IC50 > 19000 nM T38087 C13AIW 16031304 IC50 > 19000 nM T38087 CJ2XS5 16031314 IC50 = 103 nM T38087 C9LT3B 16031344 IC50 = 31 nM T38087 CEVO35 16031408 IC50 = 239 nM T38087 C0G3QB 16034760 IC50 = 250 nM T38087 CRM1P5 16351577 IC50 = 92000 nM T38087 C4T7EK 16516470 IC50 = 272 nM T38087 CB9I0W 20254879 IC50 = 770 nM T38087 CB3UK1 21453474 IC50 > 20000 nM T38087 C3WH2U 22582929 IC50 = 2010 nM T38087 CYC63Q 22582930 IC50 = 220 nM T38087 CNIW39 22582931 IC50 = 70 nM T38087 CCS4U1 22582933 IC50 = 20 nM T38087 C0DW5F 22582935 IC50 = 9 nM T38087 CA3TO2 22582936 IC50 = 8 nM T38087 CMF72I 22582975 IC50 = 39 nM T38087 CZSY32 22582976 IC50 = 303 nM T38087 CHF3C0 23828046 IC50 = 2700 nM T38087 C5JF8P 27396804 IC50 > 19000 nM T38087 CP5S9R 27532289 IC50 = 980 nM T38087 CMXA39 28825277 IC50 > 100000 nM T38087 CSO1Z6 28825295 IC50 > 100000 nM T38087 CY5UH1 29717874 IC50 = 353 nM T38087 CW9C8F 34260323 IC50 = 1880 nM T38087 CQG40E 41783892 IC50 = 2760 nM T38087 CNX30Y 43817831 IC50 = 10000 nM T38087 C8BKV6 44381234 IC50 = 44.67 nM T38087 CNI3Y5 44483163 IC50 = 39 nM T38087 CDE3H4 46952397 IC50 = 6309.57 nM T38087 CTE39K 49832752 IC50 = 51 nM T38087 CXR9G1 49833459 IC50 = 290 nM T38087 C9V5PW 49834204 IC50 > 10000 nM T38087 CU8M9C 53550548 IC50 = 93000 nM T38087 CNQ5M1 53550662 IC50 = 2100 nM T38087 CM2HE3 53554468 IC50 = 140000 nM T38087 CWF40I 56587957 IC50 = 30.9 nM T38087 C2TG1V 57378623 IC50 = 12300 nM T38087 CX17EU 57378738 IC50 = 54 nM T38087 CD3HT9 67960134 IC50 = 85.5 nM T38087 CA9VM2 68166499 IC50 > 10000 nM T38087 C4EIK5 68166523 IC50 = 1800 nM T38087 CWV26A 68166560 IC50 = 43 nM T38087 CJ9N2T 70693730 IC50 > 19000 nM T38087 C24XZF 71576800 IC50 = 52 nM T38087 CKFI57 71576801 IC50 = 39 nM T38087 C8KYW4 71576802 IC50 = 22 nM T38087 C5IS2J 71576803 IC50 = 9 nM T38087 COA6C9 71576804 IC50 = 21 nM T38087 CED5V6 71622125 IC50 = 2290.87 nM T38087 CI0GU8 71660496 IC50 = 2 nM T38087 CBJF48 71681828 IC50 = 310 nM T38087 C2LDQ3 71681829 IC50 = 150 nM T38087 C9Y0DK 71681830 IC50 = 9 nM T38087 CTOM14 71681831 IC50 = 1370 nM T38087 CO96XF 71819164 IC50 = 127 nM T38087 CMC2J4 72193935 IC50 = 26 nM T38087 CL73DQ 72549316 IC50 = 79.43 nM T38087 CX9BU6 72549541 IC50 = 19.95 nM T38087 C06VKU 72549782 IC50 = 100 nM T38087 C2U6AT 72699516 IC50 < 60 nM T38087 C3E9CI 72699517 IC50 < 60 nM T38087 CO4U3W 72699596 IC50 = 93 nM T38087 CR3ZE1 72699600 IC50 < 60 nM T38087 CJP9L5 72699677 IC50 < 60 nM T38087 C8AE1X 72699858 IC50 < 60 nM T38087 CA0X9C 72699953 IC50 < 60 nM T38087 CLQ5E2 72700032 IC50 < 60 nM T38087 CL3J2U 73056614 IC50 = 5 nM T38087 C28VSM 73292725 IC50 = 264 nM T38087 C2U3IW 73292882 IC50 = 202 nM T38087 C71ZFG 73292883 IC50 = 26 nM T38087 CPK8F7 73292884 IC50 = 89 nM T38087 C9NBU3 73293049 IC50 = 444 nM T38087 CQ3S2D 73293050 IC50 = 2320 nM T38087 CAT13U 73293051 IC50 = 12 nM T38087 C8DX4G 73293052 IC50 = 5 nM T38087 CK67DZ 73293053 IC50 = 3 nM T38087 CE14PD 73293054 IC50 = 33 nM T38087 CE4PM3 73293055 IC50 = 1 nM T38087 CK7MF5 73293210 IC50 = 138 nM T38087 C32GOR 73293211 IC50 = 134 nM T38087 C2WCT7 73293212 IC50 = 88 nM T38087 CTC35F 73293213 IC50 = 1790 nM T38087 CMUJ54 73293214 IC50 = 195 nM T38087 C7QO8W 73347342 IC50 = 180 nM T38087 CH3AT1 76280996 IC50 = 423 nM T38087 C8IT9R 76684090 IC50 = 289.8 nM T38087 CRE2U3 77050682 IC50 = 15000 nM T38087 C9VP6T 86276157 IC50 = 200 nM T38087 C3XO5D 89649815 IC50 = 2137.96 nM T38087 C83KNV 89661926 IC50 = 2230 nM T38087 CF8W2B 91928421 IC50 = 16000 nM T38087 C2XR5Q 92045137 IC50 = 160 nM T38087 CV0NZ7 105539834 IC50 = 37 nM T38087 CXNK07 110221018 IC50 = 2300 nM T38087 C5X1MJ 110221020 IC50 = 6600 nM T38087 CLZ1U3 118498201 IC50 = 0.18 nM T38087 CT78JM 118498266 IC50 = 0.17 nM T38087 C1VB9L 118507411 IC50 = 0.16 nM T38087 CI70KV 118717515 IC50 = 283 nM T38087 CRK45H 122177906 IC50 = 8100 nM T38087 C8GS6E 122177907 IC50 = 8300 nM T38087 CH3RJ2 122177909 IC50 = 910 nM T38087 CL4A3P 122177910 IC50 = 2398.83 nM T38087 CVCS41 122177963 IC50 = 467.74 nM T38087 CDX95C 122177964 IC50 = 7900 nM T38087 CYWJ91 122177965 IC50 = 330 nM T38087 CE0T1M 122182440 IC50 = 63000 nM T38087 CW05QD 122182441 IC50 = 4466.84 nM T38087 C5WI2T 122182442 IC50 = 230000 nM T38087 CD4KZ8 122182443 IC50 = 1949.84 nM T38087 CNEK61 122182444 IC50 = 758.58 nM T38087 C58TDA 122182445 IC50 = 5370.32 nM T38087 C9C2PH 122182446 IC50 = 53000 nM T38087 C02SDC 122423373 IC50 > 3000 nM T38087 CF2NO9 127037410 IC50 = 257.04 nM T38087 CV06MU 131801402 IC50 = 19 nM T38087 CV30YE 131801403 IC50 = 340 nM T38087 CWO68I 135153830 IC50 = 1060 nM T38087 CJ1OL3 135153891 IC50 = 120 nM T38087 C3RM9W 135153946 IC50 = 9.8 nM T38087 CD1R6Q 135400456 IC50 = 2200 nM T38087 C9PI7O 135402338 IC50 = 259 nM T38087 C0HQF2 135404247 IC50 = 54 nM T38087 C95RAN 135405744 IC50 = 189 nM T38087 C6FY0X 135416131 IC50 = 690 nM T38087 C6DBN7 135417258 IC50 = 128 nM T38087 CCY9H6 135417291 IC50 = 25 nM T38087 C1KBX6 135417551 IC50 = 58.9 nM T38087 C1PE8H 135417609 IC50 = 45.5 nM T38087 C47LAF 135418940 IC50 = 3.6 nM T38087 CIS9K5 135421564 IC50 = 101 nM T38087 CM5Q1Z 135430309 IC50 = 52 nM T38087 C4MW7F 135443732 IC50 = 459 nM T38087 CH14EB 135443955 IC50 = 8.7 nM T38087 C8XI3K 135448518 IC50 = 620 nM T38087 CZ9GA7 135449434 IC50 > 100000 nM T38087 CA0R7X 135452109 IC50 = 540 nM T38087 C9H1VA 135456692 IC50 = 1076 nM T38087 C8J2PC 135456762 IC50 = 10 nM T38087 C6C5ZS 135477410 IC50 = 720 nM T38087 COHR95 135478170 IC50 = 106 nM T38087 CHY9C3 135479130 IC50 = 1102 nM T38087 C83PBI 135491323 IC50 = 63095.73 nM T38087 CJO81C 135513650 IC50 = 86 nM T38087 C7G6BQ 135513721 IC50 = 87 nM T38087 CU3FW2 135566794 IC50 = 2 nM T38087 CG06FQ 135566852 IC50 = 7.5 nM T38087 C8QDG3 135566882 IC50 = 4.1 nM T38087 CVD04P 135566883 IC50 = 13 nM T38087 CNVM21 135566884 IC50 = 7.6 nM T38087 C4BFY3 135566969 IC50 = 6.7 nM T38087 C59OUK 135566970 IC50 = 21.5 nM T38087 C7K5WL 135566971 IC50 = 45 nM T38087 CN74FK 135566972 IC50 = 167 nM T38087 CRY12I 135566973 IC50 = 44 nM T38087 CU2I7X 135567125 IC50 = 0.2 nM T38087 C37PTU 135567126 IC50 = 0.1 nM T38087 CT1DZ8 135644892 IC50 = 39.7 nM T38087 C38XBR 135652704 IC50 = 19.4 nM T38087 C1G4CE 135741330 IC50 = 163 nM T38087 CG73ZN 135741844 IC50 = 148 nM T38087 CJB1I0 135741853 IC50 = 86 nM T38087 CAT50N 135741861 IC50 = 378 nM T38087 CY0M2Z 135741890 IC50 = 55 nM T38087 C2C7QU 135741891 IC50 = 75 nM T38087 C4ZGO7 135741892 IC50 = 32 nM T38087 CR97UC 135741893 IC50 = 81 nM T38087 CIK14M 135741895 IC50 = 136 nM T38087 C9UZ3W 135741897 IC50 = 22 nM T38087 CK39XZ 135741902 IC50 = 202 nM T38087 CIL7K3 135742498 IC50 = 107.15 nM T38087 CS83CJ 135905416 IC50 = 0.4786 nM T38087 C54NVS 136175126 IC50 = 0.28 nM T38087 CVH7R6 136175127 IC50 = 3.9 nM T38087 CS5PH8 136175128 IC50 = 0.19 nM T38087 CY94ZB 136215772 IC50 = 33 nM T38087 C7JEG1 136215773 IC50 = 40 nM T38087 CF7O2U 136215774 IC50 = 44 nM T38087 CFP0V5 136215897 IC50 = 5.5 nM T38087 C19ELM 136219321 IC50 = 11 nM T38087 C1VR8I 136219322 IC50 = 216 nM T38087 C2HJ0Y 136219323 IC50 = 2930 nM T38087 C6CT2H 136219324 IC50 = 62 nM T38087 C14DIO 136219325 IC50 = 41 nM T38087 C18GVR 136224209 IC50 = 6.2 nM T38087 CBQ6R1 136224211 IC50 = 2.5 nM T38087 CB19RP 136227775 IC50 = 62 nM T38087 CX3Z6W 136232682 IC50 = 78 nM T38087 CJW16C 136232684 IC50 = 64 nM T38087 CJ74VD 136232685 IC50 = 284 nM T38087 CSL45U 136232686 IC50 = 766 nM T38087 C8WOG5 136232687 IC50 = 180 nM T38087 C47HSR 136232688 IC50 = 345 nM T38087 C3D4LH 136232691 IC50 = 958 nM T38087 CZU8W3 136232694 IC50 = 4780 nM T38087 CR7Q4L 136232699 IC50 = 1030 nM T38087 CM4PB2 136236970 IC50 = 10.5 nM T38087 C50JYC 136236972 IC50 = 30 nM T38087 C1WG3C 136236974 IC50 = 21 nM T38087 CF1H5N 136236975 IC50 = 39 nM T38087 CU17IT 136236976 IC50 = 12 nM T38087 C71FDZ 136236977 IC50 = 14 nM T38087 CCL4D6 136236978 IC50 = 20 nM T38087 C9WHB4 136236979 IC50 = 3.6 nM T38087 C68GON 136236980 IC50 = 12 nM T38087 C18MSY 136236981 IC50 = 7 nM T38087 CF01JX 136236982 IC50 = 7.5 nM T38087 CYF2I1 136236983 IC50 = 700 nM T38087 C3ZW8J 136236994 IC50 = 1.5 nM T38087 CN0J1C 136236995 IC50 = 50 nM T38087 CHJ8I2 136236997 IC50 = 1.4 nM T38087 C0LB6W 136236998 IC50 = 0.5 nM T38087 CVB4D7 136237000 IC50 = 40 nM T38087 CSB3Y1 136237004 IC50 = 1.8 nM T38087 C4H8ZN 136237010 IC50 = 38 nM T38087 CW9H8J 136237302 IC50 = 23 nM T38087 CV6OL8 136237316 IC50 = 6 nM T38087 CA60VL 136237359 IC50 = 31 nM T38087 CI5FO2 136237361 IC50 = 11 nM T38087 C6JH2X 136237372 IC50 = 18 nM T38087 CAEC09 136237382 IC50 = 57 nM T38087 C4DB3K 136237396 IC50 = 16 nM T38087 CB9E1U 136239479 IC50 = 7960 nM T38087 CRWN30 136241639 IC50 = 0.4 nM T38087 CEWX52 136244045 IC50 = 35 nM T38087 CTP76D 136244148 IC50 = 63 nM T38087 CC4RQ3 136244160 IC50 = 18700 nM T38087 CR07BF 136244504 IC50 = 2 nM T38087 CHSN59 136245073 IC50 = 100 nM T38087 C2P5LK 136253145 IC50 = 14 nM T38087 C0D8MZ 136264443 IC50 = 49 nM T38087 CUPY84 136268378 IC50 = 67.6 nM T38087 CF3X4M 136372378 IC50 = 263 nM T38087 CUB67C 136404917 IC50 > 100000 nM T38087 CWH02F 136491252 IC50 = 15 nM T38087 CF80AR 136491263 IC50 = 106 nM T38087 C6T9OI 136947736 IC50 = 2.2 nM T38087 C91WJF 136947741 IC50 = 0.7 nM T38087 CFS5Z4 136947743 IC50 = 31 nM T38087 CVM4S9 136947751 IC50 = 43 nM T38087 C9UGV5 137169064 IC50 = 79.8 nM T38087 CMN5H6 137169065 IC50 = 28.6 nM T38087 CS7ZQ8 137637696 IC50 = 6.457 nM T38087 CKM58P 137638894 IC50 = 2.512 nM T38087 CA9EU4 137641940 IC50 = 199.53 nM T38087 CW1C2I 137647832 IC50 = 6.31 nM T38087 CETG37 137652318 IC50 = 316.23 nM T38087 C72DEL 137657753 IC50 = 25.12 nM T38087 CW7GD8 137659255 IC50 = 19.95 nM T38087 C4R7VI 137701512 IC50 = 10.6 nM T38087 CWLV03 138594154 IC50 = 18.7 nM T38087 CDW5N1 138594164 IC50 = 11.1 nM T38087 CSK82I 138594166 IC50 = 6.4 nM T38087 CD1M0Y 138594171 IC50 = 23.4 nM T38087 C9QYJ3 138594172 IC50 = 20.2 nM T38087 C1XSH7 138594194 IC50 = 39.2 nM T38087 C4JO9N 138594198 IC50 = 6.1 nM T38087 C7I1CT 138594235 IC50 = 21.4 nM T38087 CVI5N9 138594242 IC50 = 13.5 nM T38087 CS8U3T 138594273 IC50 = 17.1 nM T38087 CYR32Z 138594277 IC50 = 7 nM T38087 CNSV30 138594278 IC50 = 21.2 nM T38087 C1C2AS 138594290 IC50 = 33.3 nM T38087 C34OCY 138594292 IC50 = 8.5 nM T38087 CUA1E8 138594320 IC50 = 4.7 nM T38087 CGE6Q5 138594327 IC50 = 12.4 nM T38087 C0RST4 138594360 IC50 = 21 nM T38087 C4K7MW 138594363 IC50 = 6.8 nM T38087 CNW2O9 138594369 IC50 = 5.3 nM T38087 C3F7MV 138594378 IC50 = 10.4 nM T38087 C6YU8S 138594385 IC50 = 15.6 nM T38087 C48AGS 138594414 IC50 = 20.7 nM T38087 CA49EZ 138594436 IC50 = 14.6 nM T38087 CL6EV4 138594465 IC50 = 9.9 nM T38087 CJL05F 138594467 IC50 = 18.5 nM T38087 CX4SL6 138594472 IC50 = 2.8 nM T38087 C3E5IU 138594491 IC50 = 27.6 nM T38087 C13EVQ 138594498 IC50 = 35.7 nM T38087 C4L9XQ 138594506 IC50 = 26.9 nM T38087 CKF1W3 138594528 IC50 = 14.4 nM T38087 C98NUR 138594556 IC50 = 6.2 nM T38087 CDZ43N 138594558 IC50 = 10.7 nM T38087 CLD3J5 138594570 IC50 = 12.3 nM T38087 CWVO67 138594578 IC50 = 16.4 nM T38087 C6QD2W 138594607 IC50 = 4.9 nM T38087 CP6Y5L 138594610 IC50 = 10.2 nM T38087 CSQJ12 138594627 IC50 = 3.4 nM T38087 CEOJ61 138594628 IC50 = 4.7 nM T38087 CU4O9K 138594631 IC50 = 7.1 nM T38087 C0A4FG 138594645 IC50 = 12 nM T38087 CN3U9X 138594667 IC50 = 9.5 nM T38087 CQK29G 138594732 IC50 = 5.8 nM T38087 CCU4I1 138594747 IC50 = 7.5 nM T38087 C1KWY7 138594763 IC50 = 13.4 nM T38087 C9HR2J 138594785 IC50 = 18.3 nM T38087 CP4NF9 138594790 IC50 = 25.1 nM T38087 CF74SW 138594809 IC50 = 26.8 nM T38087 CF7ZR5 138594952 IC50 = 15.1 nM T38087 CW5E6D 138594964 IC50 = 7.6 nM T38087 CURM89 138594969 IC50 = 17 nM T38087 C72QVS 138595093 IC50 = 29.3 nM T38087 CX7PZ5 141639950 IC50 > 100000 nM T38087 C8I9CD 142613964 IC50 = 3.3 nM T38087 C5SG1U 145957836 IC50 = 576 nM T38087 C6HOA3 145972257 IC50 = 2800 nM T38087 CA65UC 145974539 IC50 = 953 nM T38087 COB76P 145989667 IC50 = 56 nM T38087 CPY72O 153951026 IC50 = 13 nM T38087 CWV08R 155511996 IC50 = 3476 nM T38087 CZ78CA 155513337 IC50 = 6417 nM T38087 CRX36I 155515281 IC50 = 5.5 nM T38087 CC9J2N 155516254 IC50 = 13 nM T38087 C6EJ7I 155518170 IC50 = 6984 nM T38087 CIC9H8 155518184 IC50 = 10.5 nM T38087 C1DL6E 155518640 IC50 = 148 nM T38087 CGKW04 155520067 IC50 > 20000 nM T38087 CHV6T4 155521523 IC50 = 2.3 nM T38087 CUM52X 155522687 IC50 = 2.6 nM T38087 CEP6Y5 155528458 IC50 = 36.4 nM T38087 C91IPT 155529963 IC50 = 12.5 nM T38087 CA9XP1 155531429 IC50 = 29.8 nM T38087 CL2PO4 155532179 IC50 = 11.7 nM T38087 C09PYD 155532212 IC50 = 112 nM T38087 C4JPD1 155532717 IC50 = 49.1 nM T38087 CZL4U1 155534087 IC50 = 32.4 nM T38087 CV2MX1 155535415 IC50 = 49.7 nM T38087 CY8RJ7 155537249 IC50 = 198 nM T38087 CWM48X 155538013 IC50 = 65.5 nM T38087 CU65VW 155540828 IC50 = 258 nM T38087 CZN0O1 155541146 IC50 = 9336 nM T38087 CYWG48 155541643 IC50 > 1000 nM T38087 C9INM1 155543325 IC50 = 11.8 nM T38087 CG0J7F 155545779 IC50 = 8.8 nM T38087 CO0E8F 155549220 IC50 = 4.8 nM T38087 CD5C9R 155550189 IC50 > 20000 nM T38087 C4P3QD 155553178 IC50 = 26 nM T38087 CIYH06 155556919 IC50 = 5345 nM T38087 CXAJ25 155557028 IC50 = 73.6 nM T38087 CWH8D0 155561438 IC50 = 12.2 nM T38087 C46UYI 155562058 IC50 = 4386 nM T38087 COH6X1 155564702 IC50 = 8.2 nM T38087 D00RIX 5280443 IC50 = 2951.21 nM T38087 D00TUB 135471356 IC50 = 219 nM T38087 D03BQJ 688829 IC50 = 190 nM T38087 D04WDX 4858 IC50 = 219 nM T38087 D06NKJ 135439437 IC50 = 1029 nM T38087 D07BPT 135457978 IC50 = 30 nM T38087 D0B2WX 135407310 IC50 = 12 nM T38087 D0E5EW 135531482 IC50 = 41 nM T38087 D0G5VD 135492389 IC50 = 191 nM T38087 D0GA0Y 135463623 IC50 = 3.3 nM T38087 D0O6WW 135528341 IC50 = 180 nM T38087 D0OF1I 135417274 IC50 = 863 nM T38087 D0S0RK 10680 IC50 = 140 nM T38087 D0Y1MH 135471354 IC50 = 3 nM T38087 D0YJ3Q 5322065 IC50 = 870 nM T32247 C1IY0P 56944164 Ki = 3200 nM T32247 CY78NF 73345422 Ki = 2569 nM T32247 CJ73DQ 73346943 Ki = 195 nM T32247 C6S3MN 73351529 Ki = 0.05 nM T32247 D00JEO 73346944 Ki = 0.051 nM T32247 D03CEP 73348438 Ki = 400 nM T32247 D03DPD 73356077 Ki = 0.56 nM T32247 D05AIM 73346940 Ki = 0.069 nM T32247 D05MSG 44593666 Ki > 5000 nM T32247 D08URJ 73351527 Ki = 42.5 nM T32247 D0A8VZ 73352989 Ki = 0.069 nM T32247 D0G0WP 73350025 Ki = 5.28 nM T32247 D0J7CK 73351528 Ki = 0.023 nM T32247 D0Y0NM 73354513 Ki > 2500 nM T03279 D0E6XR 3062316 IC50 > 20000 nM T03279 D0EG1I 9926791 IC50 > 10000 nM T03279 D0R0MW 5329102 IC50 = 183.9 nM T03279 D05PZB 135398495 IC50 = 1 nM T03279 D0E3TC 44259 IC50 = 0.124 nM T03279 D03BNU 59604787 IC50 > 10000 nM T03279 CO7J0B 587331 IC50 = 13180 nM T03279 CY13FW 644243 IC50 = 15 nM T03279 CA40OY 834921 IC50 = 1060 nM T03279 CHTL73 899653 IC50 = 480 nM T03279 CU3YF7 902492 IC50 = 2880 nM T03279 CSM95Y 1160249 IC50 = 320 nM T03279 CUJ3H4 1202309 IC50 = 17000 nM T03279 C4FL7C 1225079 IC50 = 9990 nM T03279 CYL9O2 1225114 IC50 = 1680 nM T03279 COA87I 2731384 IC50 = 950 nM T03279 CRI4S0 2978413 IC50 = 1380 nM T03279 CVQ13D 3139616 IC50 = 3470 nM T03279 CHJ78U 3274711 IC50 = 15140 nM T03279 C8BDV2 3592486 IC50 = 5500 nM T03279 CE97MX 4164840 IC50 = 1580 nM T03279 CKCH09 4668168 IC50 = 7040 nM T03279 CZ03SJ 5476622 IC50 = 3470 nM T03279 CDK3J0 5703619 IC50 = 1.6 nM T03279 C4YJ3C 5714584 IC50 = 2720 nM T03279 CZ74AJ 6164317 IC50 = 1510 nM T03279 C62USN 6164860 IC50 = 2020 nM T03279 C2PGU4 9572071 IC50 = 14000 nM T03279 CA3V0T 9572240 IC50 = 5660 nM T03279 C1DJ6B 9572244 IC50 = 3130 nM T03279 C73SQF 9572245 IC50 = 3000 nM T03279 CJR60A 9572531 IC50 = 970 nM T03279 C7GBL9 9572533 IC50 = 3760 nM T03279 C8P3DE 9572535 IC50 = 2800 nM T03279 C6MU5H 9572537 IC50 = 44800 nM T03279 CXZK43 9572545 IC50 = 5930 nM T03279 CDF2S5 9572547 IC50 = 13930 nM T03279 CXI68F 9572620 IC50 = 5850 nM T03279 CSG4X7 9572624 IC50 = 4530 nM T03279 CIFU15 9572626 IC50 = 17500 nM T03279 CK2I4R 9572632 IC50 = 98500 nM T03279 C7OZ6U 9572657 IC50 = 6430 nM T03279 CU30ZL 9572659 IC50 = 5970 nM T03279 C6NGW1 9572661 IC50 = 13250 nM T03279 CRA10N 9572663 IC50 = 20950 nM T03279 C7J4HC 9572736 IC50 = 3580 nM T03279 CJ2EP9 9999648 IC50 = 2000 nM T03279 CINF40 10073694 IC50 = 640 nM T03279 CFIE04 10459196 IC50 = 89 nM T03279 C0APW4 11422034 IC50 = 10000 nM T03279 CXBU49 11502255 IC50 = 76000 nM T03279 CTG83F 11539329 Ki > 7400 nM T03279 CACS26 11561968 Ki > 2000 nM T03279 CMIL86 11590363 Ki > 7400 nM T03279 C9T6SC 11640926 Ki = 3300 nM T03279 CU0E8O 11690457 Ki > 2000 nM T03279 CP5W1H 11964005 IC50 = 170 nM T03279 CA1PQ3 15604675 IC50 = 730 nM T03279 C6OA2P 15604847 IC50 = 210 nM T03279 CFPW41 16007116 Ki > 7400 nM T03279 C9TU1O 16046126 IC50 > 1000 nM T03279 CCQ1W9 16099270 IC50 = 100000 nM T03279 CB04TO 16099272 IC50 = 100000 nM T03279 CHQL75 16099330 IC50 = 83000 nM T03279 C5VPH9 16129448 IC50 = 83 nM T03279 CGA1H4 16662748 IC50 = 250 nM T03279 C6QH4P 20299668 IC50 > 100000 nM T03279 C1S9ZB 20299672 IC50 > 100000 nM T03279 C1XLM5 24204009 IC50 = 20500 nM T03279 CMU75L 24204554 IC50 = 26500 nM T03279 CSM03X 24204556 IC50 = 79000 nM T03279 CB4Y6K 24204558 IC50 = 7320 nM T03279 C1TR9Z 24205072 IC50 = 94000 nM T03279 C5GS0O 24205074 IC50 = 2890 nM T03279 C7YG1N 24759534 IC50 = 260 nM T03279 C0MO8J 24800837 IC50 = 18000 nM T03279 CUZP05 24901001 IC50 > 100000 nM T03279 CLZ23U 24951610 IC50 = 1300 nM T03279 C2KY1G 25094210 IC50 = 1306 nM T03279 CGT1W6 25144294 IC50 = 360 nM T03279 CU7VR0 25144732 IC50 = 180 nM T03279 C6BWZ8 25145145 IC50 > 100 nM T03279 C78YWA 25145716 IC50 = 260 nM T03279 CEM7A3 39222210 IC50 = 2500 nM T03279 CU0MG3 44141269 IC50 = 4 nM T03279 C40JYN 44143549 IC50 = 350 nM T03279 CNA95E 44143558 IC50 = 240 nM T03279 CH2F9K 44143559 IC50 = 2200 nM T03279 C04QTA 44143560 IC50 = 1800 nM T03279 CIH05K 44143561 IC50 = 1200 nM T03279 CO6HU7 44178069 IC50 = 1100 nM T03279 COPG94 44427519 IC50 > 10000 nM T03279 C3VRO9 44557921 IC50 > 10000 nM T03279 CG7CV6 44565316 IC50 = 430000 nM T03279 CF90OX 44576212 IC50 = 39000 nM T03279 CY3HW5 46224684 IC50 = 4000 nM T03279 CLS29B 46872626 IC50 > 10000 nM T03279 C1NKE3 46905987 IC50 = 48 nM T03279 C4R5CJ 49864389 IC50 = 1700 nM T03279 CW53JF 49864404 IC50 = 20 nM T03279 CQ81GN 51029632 IC50 = 1230 nM T03279 C5ME1Y 51029719 IC50 = 1600 nM T03279 CD3P9O 51029720 IC50 = 270 nM T03279 COIX20 51029721 IC50 = 620 nM T03279 CN3IR4 51029723 IC50 = 710 nM T03279 C1XP3S 51029811 IC50 = 1770 nM T03279 CC0I6L 51029813 IC50 = 1500 nM T03279 CXA03W 52920796 IC50 > 100 nM T03279 C50QPW 52938516 IC50 = 7 nM T03279 CG2F0P 52938644 IC50 = 5 nM T03279 CGI5U6 52939498 IC50 = 4 nM T03279 CAT53K 53247439 IC50 = 1 nM T03279 CO5N8J 53247559 IC50 = 12 nM T03279 CM29QI 53247560 IC50 = 2 nM T03279 CPK70S 53247680 IC50 = 14 nM T03279 CE8OY2 53317913 IC50 > 100 nM T03279 C0SWH5 53348216 IC50 > 40000 nM T03279 CXV2G6 54770686 IC50 = 8260 nM T03279 C0C7JF 54770689 IC50 > 100000 nM T03279 CES4B3 54770691 IC50 = 86000 nM T03279 C6Z2VS 54770693 IC50 = 3930 nM T03279 C3ZVT2 54770915 IC50 = 8550 nM T03279 CZ3C1P 54770917 IC50 > 100000 nM T03279 C1IX4N 54771375 IC50 > 100000 nM T03279 CME94T 54771590 IC50 = 12000 nM T03279 C5GPT9 54771592 IC50 = 10150 nM T03279 CQY26A 54771820 IC50 > 100000 nM T03279 C1TWQ3 54771822 IC50 = 7800 nM T03279 CYX98P 56834879 IC50 = 4 nM T03279 CK0WS8 56834880 IC50 = 200 nM T03279 CY83FV 56835180 IC50 = 19 nM T03279 CB5XP4 56840684 IC50 = 750 nM T03279 CQ57PE 57345536 IC50 = 68 nM T03279 CI82KP 57390271 IC50 > 100000 nM T03279 CHU67R 57390273 IC50 = 30670 nM T03279 CS58YJ 57390566 IC50 = 45 nM T03279 CREQ53 57390567 IC50 = 180 nM T03279 CK7Q2U 57390653 IC50 = 4600 nM T03279 CFG98J 57390654 IC50 = 53 nM T03279 C6AP5W 57391812 IC50 > 10000 nM T03279 C4CIW6 57391813 IC50 = 86 nM T03279 CN6C1Q 57392344 IC50 = 1930 nM T03279 CEUL82 57392345 IC50 = 400 nM T03279 CV8Z3C 57392346 IC50 = 21 nM T03279 CFU03W 57392455 IC50 = 1700 nM T03279 CNDW76 57392456 IC50 = 68 nM T03279 C61CIX 57393506 IC50 = 160 nM T03279 CE8T5V 57393795 IC50 = 607.1 nM T03279 CM6F0O 57393798 IC50 = 6030 nM T03279 C7C1ZG 57394084 IC50 = 9100 nM T03279 CV6F2R 57394085 IC50 = 26 nM T03279 CN01TQ 57394160 IC50 = 240 nM T03279 CN4B2W 57394161 IC50 = 410 nM T03279 CBP29W 57394162 IC50 = 3300 nM T03279 C3A1DV 57394163 IC50 = 367 nM T03279 CGU57X 57394413 IC50 = 56730 nM T03279 CZ2NE3 57395227 IC50 = 6 nM T03279 C2YUD9 57395253 IC50 = 7 nM T03279 CT9L8D 57395512 IC50 > 100000 nM T03279 C2VYZ5 57395514 IC50 > 100000 nM T03279 CGU6C4 57395516 IC50 = 53750 nM T03279 C5KS6T 57395518 IC50 > 100000 nM T03279 C81JSP 57395520 IC50 > 100000 nM T03279 COD4J5 57395855 IC50 = 970 nM T03279 C4Z5FG 57395945 IC50 > 10000 nM T03279 CQ6Y4G 57397344 IC50 = 2150 nM T03279 CIG5D8 57397643 IC50 = 34 nM T03279 CMWC20 57397644 IC50 = 2200 nM T03279 CGX4M2 57397731 IC50 = 43 nM T03279 CHO1L5 57397732 IC50 = 34 nM T03279 C8TN0X 57398716 IC50 = 10 nM T03279 CS09AU 57398752 IC50 = 18 nM T03279 CSGJ63 57398759 IC50 = 27 nM T03279 CQG54I 57398793 IC50 = 11 nM T03279 C0HQ1R 57399029 IC50 > 100000 nM T03279 CV2GB8 57399310 IC50 = 871 nM T03279 C9HGU7 57399311 IC50 > 10000 nM T03279 CMCZ72 57399312 IC50 = 52 nM T03279 C3KOR1 57399398 IC50 = 2500 nM T03279 CUJO50 57399399 IC50 = 540 nM T03279 CD4W5E 57399400 IC50 > 10000 nM T03279 C5JI1M 57400390 IC50 = 180 nM T03279 C48QMJ 57400429 IC50 = 61 nM T03279 CA7P1L 57400430 IC50 = 4 nM T03279 C6PCR8 57400465 IC50 = 26 nM T03279 CLZ19B 57400466 IC50 = 13 nM T03279 CU82DZ 57400761 IC50 > 100000 nM T03279 CF5LW8 57400763 IC50 > 100000 nM T03279 CVE76G 57401078 IC50 > 10000 nM T03279 C49RWO 57401079 IC50 = 270 nM T03279 CMH67I 57401161 IC50 = 41 nM T03279 CMTE87 57401162 IC50 = 1100 nM T03279 CN94VT 57401163 IC50 = 93 nM T03279 CE60BZ 57402527 IC50 > 100000 nM T03279 CECL89 57402533 IC50 = 18500 nM T03279 CRE6H0 57402838 IC50 = 6000 nM T03279 C7LKZ3 57402839 IC50 = 220 nM T03279 C07JNH 57402840 IC50 > 10000 nM T03279 C6ST9X 57402925 IC50 > 1000 nM T03279 CO95QU 57403971 IC50 = 21 nM T03279 C6BPR2 58985201 IC50 = 27000 nM T03279 CP9A8T 59503659 IC50 = 6800 nM T03279 C1MA6J 59503711 IC50 = 4300 nM T03279 CX29EU 59503744 IC50 = 7700 nM T03279 CXJ63M 59603829 IC50 = 380 nM T03279 CQEU96 59603842 IC50 < 1 nM T03279 C1MR8Q 60097495 IC50 > 1000 nM T03279 CNPZ43 60150536 IC50 = 252 nM T03279 C4EW8A 60150537 IC50 = 869 nM T03279 CTHS89 60150538 IC50 = 1920 nM T03279 CK6WO0 66552478 IC50 < 10000 nM T03279 C37NKO 67129970 IC50 = 9810 nM T03279 CG6XQ3 67161715 IC50 = 24 nM T03279 CNXU89 67162253 IC50 = 248 nM T03279 CV63UL 67240318 IC50 > 10000 nM T03279 C7GRV2 68755406 IC50 > 10000 nM T03279 C5DGR9 69036886 IC50 = 692 nM T03279 CMFU48 70689587 IC50 = 1130 nM T03279 C9M3GH 70691716 IC50 = 493 nM T03279 CU36AQ 70695907 IC50 = 356 nM T03279 CUZ4C7 70695908 IC50 = 1430 nM T03279 CKT60L 71455860 Ki = 630 nM T03279 CSE1U7 71511480 IC50 = 8590 nM T03279 C1YB8V 71527472 IC50 = 1510 nM T03279 CTCK49 71527473 IC50 = 480 nM T03279 CU62XK 71680549 IC50 = 2490 nM T03279 C3GN9B 71718779 IC50 = 20 nM T03279 CBZC56 73010393 IC50 = 5 nM T03279 C1HW4B 89735655 IC50 = 47 nM T03279 CAU45T 91971978 IC50 > 30000 nM T03279 C0VIF3 118704762 IC50 = 4 nM T03279 CKAZ73 118721541 IC50 = 8930 nM T03279 CUV59P 122186015 IC50 = 60 nM T03279 CU94BL 122186016 IC50 = 130 nM T03279 C7P5RV 122186017 IC50 = 2100 nM T03279 C46ROU 122186018 IC50 = 780 nM T03279 CG1WL0 122186019 IC50 = 32 nM T03279 C9L1FX 122186020 IC50 = 46 nM T03279 C9P3WB 122186021 IC50 = 4 nM T03279 C8ZYK2 122186022 IC50 = 5 nM T03279 C26XBR 122186023 IC50 = 18 nM T03279 C15SDH 122186024 IC50 = 4 nM T03279 COZW89 122186025 IC50 = 94 nM T03279 C2GU9S 122186026 IC50 = 7 nM T03279 C54NHE 122186027 IC50 = 8 nM T03279 C73FHA 122186028 IC50 = 20 nM T03279 C2DZB3 122186029 IC50 = 6 nM T03279 C86TBG 122186030 IC50 = 80 nM T03279 C9P5BZ 122186031 IC50 = 4800 nM T03279 CW4FS1 122186114 IC50 = 6 nM T03279 CI52DY 122186115 IC50 = 14 nM T03279 COF9H4 122186116 IC50 = 22 nM T03279 CXH91E 122186117 IC50 = 6 nM T03279 C4RT7V 122186118 IC50 = 10 nM T03279 CEL4N7 122186119 IC50 = 13 nM T03279 CQ8R2O 122186120 IC50 = 23 nM T03279 CW8F2P 122186121 IC50 = 20 nM T03279 CS4OW8 135400873 Ki > 2000 nM T03279 CPY35Q 135411960 IC50 = 16180 nM T03279 CE42LA 135453602 IC50 = 14450 nM T03279 CYMW12 135567074 IC50 = 20 nM T03279 CW72QO 135580408 IC50 = 11400 nM T03279 CFAD48 135611170 Ki > 2000 nM T03279 CT92RP 136088964 IC50 = 3030 nM T03279 CAK0W2 136110946 IC50 = 6 nM T03279 CLIM07 136110947 IC50 = 53 nM T03279 C3J7OC 136110948 IC50 = 150 nM T03279 CK38HO 137125250 IC50 = 50 nM T03279 CBE35D 137125251 IC50 = 180 nM T03279 CI1E8V 137634241 IC50 > 10000 nM T03279 CDNC31 145967951 IC50 = 180 nM T03279 C8DNZ1 145979228 IC50 = 240 nM T03279 CU7S1Q 145980512 IC50 = 2 nM T03279 CF3KI9 145984908 IC50 = 500 nM T03279 CTW7F0 145984931 IC50 = 800 nM T03279 C03PYD 145986466 IC50 = 0.3 nM T03279 CD8Z6O 145986826 IC50 = 2 nM T03279 CO4P3E 145989941 IC50 = 38 nM T03279 CK9U2I 145990304 IC50 = 810 nM T03279 CV2NB6 145991585 IC50 = 1100 nM T03279 C1S8WN 145993273 IC50 = 1900 nM T03279 C2MD1Q 155513187 IC50 > 10000 nM T03279 D00ERW 44444843 Ki > 7368 nM T03279 D00HVA 11624601 Ki > 7400 nM T03279 D09PTP 57325421 IC50 = 13 nM T03279 D0C2GE 67161540 IC50 = 3 nM T03279 D0CM6T 11314340 Ki = 580 nM T03279 D0M5FF 5083 IC50 = 10 nM T03279 D0ME9B 46868971 IC50 = 330 nM T03279 D0Q3NG 11715520 Ki > 7400 nM T03279 D0S7IE 11658882 Ki > 7400 nM T03279 D0U3NI 53246941 IC50 = 1 nM T85605 D01UTL 2995 IC50 = 350 nM T85605 D04JCN 47811 IC50 = 385 nM T85605 D04WFD 4543 IC50 = 170 nM T85605 D06ZUK 3696 IC50 = 44 nM T85605 D0H6QU 6005 IC50 = 4500 nM T85605 D0K7WK 4595 Ki > 10000 nM T85605 D0R6RO 4184 IC50 > 5000 nM T85605 D0W9ZF 3086401 IC50 = 2300 nM T85605 D0Y5UG 2160 IC50 = 44 nM T85605 D0ZS8P 2801 IC50 = 5 nM T85605 D0Z2MB 6918107 Ki > 10000 nM T85605 CJ0B9F 3158 IC50 = 200 nM T85605 CJF27B 17654 IC50 = 630 nM T85605 CG5T8J 19219 IC50 = 220 nM T85605 CK15QR 21180 IC50 = 1000 nM T85605 C80INW 36431 IC50 > 1000 nM T85605 CI30OT 193459 IC50 = 151000 nM T85605 C78LRZ 13140993 IC50 = 40700 nM T85605 C9GHK1 13141004 IC50 = 933000 nM T85605 C1LO5W 14687338 IC50 = 660693.45 nM T85605 C0E1DB 44278537 IC50 = 40800 nM T85605 C6VB8R 44348574 IC50 = 720 nM T85605 C3B8VC 44383444 IC50 = 2240 nM T85605 CW4E2J 46220521 IC50 > 10000 nM T85605 CY92LZ 53310757 Ki > 1000 nM T85605 C8GQK9 73350823 Ki = 1270 nM T85605 D0YG1E 68847 IC50 = 26 nM T74238 D00QET 5281040 IC50 > 10000 nM T74238 D05DVP 5717 IC50 = 7397 nM T74238 D08QIP 4887 IC50 = 3620 nM T74238 D0U5YM 46830962 IC50 = 25 nM T74238 CA5OL4 5311184 IC50 = 43000 nM T74238 CO8KI0 11191817 IC50 = 2.3 nM T74238 CS0J3E 11227280 IC50 = 16 nM T74238 CFMP93 11249398 IC50 = 30 nM T74238 CA5G8V 11261220 IC50 = 3.4 nM T74238 CGHR62 11284237 IC50 = 17 nM T74238 CC9VH6 11307317 IC50 = 0.62 nM T74238 CK9ST2 11353238 IC50 = 15 nM T74238 C91OUF 11387037 IC50 = 55 nM T74238 C3TL2O 11398475 IC50 = 0.87 nM T74238 CW8D7G 11398820 IC50 = 0.49 nM T74238 CC1S3B 11455387 IC50 = 0.31 nM T74238 C69TXN 11713438 IC50 = 6 nM T74238 CWH9Q3 11853184 IC50 = 25 nM T74238 C45JZF 23124563 IC50 = 890 nM T74238 CKGH56 23124623 IC50 = 68 nM T74238 CROH42 23124629 IC50 = 890 nM T74238 C3HYZ8 23124664 IC50 = 5.7 nM T74238 CLW5A4 23124672 IC50 = 1800 nM T74238 C1L5NF 23124680 IC50 = 5.7 nM T74238 CDCT78 23124707 IC50 = 16 nM T74238 C9NAV8 23124716 IC50 = 16 nM T74238 CE8S9N 23124741 IC50 = 1500 nM T74238 CXQ38G 23124775 IC50 = 290 nM T74238 CRW4V9 23663996 IC50 = 27000 nM T74238 CSB4R8 46830677 IC50 = 3.6 nM T74238 C9BHQ2 46830961 IC50 = 12 nM T74238 C9DXV5 46830963 IC50 = 13 nM T74238 C9BT3C 46834997 IC50 = 5.5 nM T74238 C3OD2Q 46835000 IC50 = 8.8 nM T74238 C4FGC6 54677430 IC50 = 7700 nM T74238 C28RDF 54746913 IC50 = 4500 nM T74238 CLGZ72 66739117 IC50 = 5.1 nM T74238 CJ7PE4 68695885 IC50 = 25 nM T74238 C2TW7S 71654671 IC50 = 7500 nM T74238 C21QBY 71654672 IC50 = 250 nM T74238 C2DCQ4 87131159 IC50 = 2.2 nM T74238 CC01GT 90871050 IC50 = 4600 nM T74238 C0B3PZ 118716774 IC50 = 3600 nM T74238 C81NVL 118716775 IC50 = 5200 nM T74238 CSTV67 118716776 IC50 = 3700 nM T74238 CHM06D 118716777 IC50 = 170 nM T74238 C8OAM0 118728613 IC50 = 4300 nM T74238 C2E5LC 118729613 IC50 = 410 nM T74238 CHV59E 118729614 IC50 = 370 nM T74238 CI48HX 118729615 IC50 = 75 nM T74238 CU8GO5 122183681 IC50 = 23 nM T74238 C57LAY 122183682 IC50 = 2.1 nM T74238 CD2X9M 122183683 IC50 = 14 nM T74238 CBZT62 122183684 IC50 = 4.6 nM T74238 CXY1J3 122183685 IC50 = 4.7 nM T74238 C8JPS5 122183686 IC50 = 15 nM T74238 C9GY0M 122183687 IC50 = 1 nM T74238 C7LR4C 122183688 IC50 = 3.7 nM T74238 C3SBE6 122183689 IC50 = 1.5 nM T74238 CI83YC 122183690 IC50 = 7.2 nM T74238 C6SP3V 122183751 IC50 = 0.89 nM T74238 CIWZ15 122183752 IC50 = 5.7 nM T74238 CMV47L 122183753 IC50 = 0.88 nM T74238 C25ETG 122183754 IC50 = 96 nM T74238 CC91EO 122183755 IC50 = 78 nM T74238 CH4K5P 122183756 IC50 = 22 nM T74238 C3DML9 122183757 IC50 = 55 nM T74238 C0IMN8 122183758 IC50 = 15 nM T74238 C9YGC0 122183759 IC50 = 248 nM T74238 CA7P1R 122183760 IC50 = 60 nM T74238 CFD79M 122183761 IC50 = 30 nM T74238 CV9G8Y 122183762 IC50 = 31 nM T74238 C1GI5T 122183763 IC50 = 48 nM T74238 C1IQ0H 127043048 IC50 > 100000 nM T74238 C0WU9P 127043049 IC50 > 100000 nM T74238 CA0V8Q 127043050 IC50 = 58000 nM T74238 CUQL23 127043053 IC50 = 36000 nM T74238 CW84IQ 127043233 IC50 > 100000 nM T74238 CW5PI4 127043236 IC50 = 23000 nM T74238 CFB30X 127043237 IC50 = 50000 nM T74238 C1A0OU 127043241 IC50 > 100000 nM T74238 COHV05 127043242 IC50 = 87000 nM T74238 CM78QW 127043243 IC50 > 100000 nM T74238 CU79CR 127043244 IC50 = 46000 nM T74238 CYL20V 127043247 IC50 = 76000 nM T74238 CXA12T 127043248 IC50 = 46000 nM T74238 CSJF19 127043252 IC50 > 100000 nM T74238 C3ULM6 127043253 IC50 > 100000 nM T74238 CT6Y3D 127043406 IC50 > 100000 nM T74238 CF42NI 127043407 IC50 > 100000 nM T74238 CP5Q0G 127043408 IC50 > 100000 nM T74238 C39QTB 127043409 IC50 > 100000 nM T74238 C6CY1T 127043410 IC50 > 100000 nM T74238 C0X9QH 127043411 IC50 > 100000 nM T74238 CD89CS 127043617 IC50 > 100000 nM T74238 CM84GW 127043618 IC50 = 15000 nM T74238 CP0D1Z 127044872 IC50 > 100000 nM T74238 C9PS6W 127045334 IC50 > 100000 nM T74238 CS2T5L 127045343 IC50 > 100000 nM T74238 D05CNT 5311015 IC50 = 300 nM T74238 D06AYN 10438479 IC50 = 3.8 nM T74238 D09JQU 53394034 IC50 = 53 nM T09742 D0GY5Z 2244 IC50 = 36000 nM T09742 C74CAT 11948653 IC50 = 3300 nM T09742 C4Q8IB 15091141 IC50 = 25000 nM T09742 CFD92K 15091142 IC50 = 20000 nM T09742 COB31G 15091144 IC50 = 21000 nM T09742 CR2A3K 25197522 IC50 = 20000 nM T09742 C1I3NH 25197523 IC50 = 18000 nM T09742 C8Q4HB 25197524 IC50 = 28000 nM T09742 C08FRK 44565323 IC50 = 18000 nM T09742 C2HR4B 44565324 IC50 = 22000 nM T09742 CFR3X5 132556065 IC50 = 31900 nM T09742 C5RPG2 132556066 IC50 = 26300 nM T09742 CF5H9U 132556067 IC50 = 19700 nM T09742 C26FMU 132556068 IC50 = 34800 nM T09742 CFW1R7 132556069 IC50 = 22900 nM T09742 CS57DY 132556070 IC50 = 9900 nM T09742 CW92OK 132556071 IC50 = 19000 nM T09742 C8VWK4 132556072 IC50 > 50000 nM T09742 C6KYH3 132556073 IC50 > 50000 nM T09742 CVC28R 132556074 IC50 > 50000 nM T09742 C4O9UW 132556075 IC50 = 26900 nM T09742 C94XPJ 134130441 IC50 = 3100 nM T09742 CR0GK9 134131239 IC50 = 2400 nM T09742 CP25ID 134131254 IC50 = 11600 nM T09742 CJ32UR 134131405 IC50 = 7800 nM T13726 D02DGU 444795 EC50 > 0.001 nM T13726 D0G2MW 446284 Ki = 7632 nM T13726 D0G3PI 449171 EC50 = 1.5 nM T13726 D0N0RU 82146 EC50 = 2.7 nM T13726 D0Q5XX 445580 Ki = 6292 nM T13726 D0Z5IU 1548887 IC50 = 82900 nM T13726 D06QXI 9863342 EC50 = 1.5 nM T13726 D08JAC 5288209 Ki > 2200 nM T13726 D09DJC 9863341 EC50 = 0.2 nM T13726 D08GRF 5287705 Ki = 4.6 nM T13726 D09YUQ 127019 EC50 = 34 nM T13726 D0YO4D 3922 Ki = 3 nM T13726 CRI78W 94391 EC50 = 42000 nM T13726 CX90MS 128016 Ki = 1900 nM T13726 C3NS4E 132775 EC50 = 170 nM T13726 C1E2FR 442048 EC50 = 26000 nM T13726 CZ8WQ4 584660 EC50 = 17000 nM T13726 CD3P5S 585022 EC50 = 28000 nM T13726 CXK08W 585035 EC50 = 40000 nM T13726 CZ7K5V 585049 EC50 = 7800 nM T13726 CT30JZ 585603 EC50 = 29000 nM T13726 C9JFT3 661071 EC50 = 9900 nM T13726 CMF7L1 737267 EC50 > 30000 nM T13726 CDVJ42 767163 EC50 > 30000 nM T13726 CWM95S 843040 EC50 = 16000 nM T13726 C5T2PS 843045 EC50 = 6700 nM T13726 CUHQ27 997606 EC50 = 24000 nM T13726 CZO04Y 1163179 IC50 = 12000 nM T13726 C30YVK 1169819 IC50 = 12000 nM T13726 C1ZX7V 1205382 Ki = 1500 nM T13726 C9OUE2 1269478 Ki = 7400 nM T13726 C5UJF1 1637033 EC50 = 21000 nM T13726 CG3WZ4 2063265 EC50 > 30000 nM T13726 C0XK6A 2194734 EC50 = 21000 nM T13726 CG9DK0 2295706 IC50 = 4800 nM T13726 CSH2V8 2758079 EC50 = 15500 nM T13726 C4XZ0V 2758080 EC50 = 9300 nM T13726 CM60VP 2758604 EC50 = 9600 nM T13726 C1UT6Y 2758738 EC50 = 22500 nM T13726 C51INO 2886165 IC50 = 18000 nM T13726 CI8NO1 3025917 EC50 = 770 nM T13726 C78QSL 3025918 EC50 = 280 nM T13726 CQ40OB 3025919 EC50 = 54 nM T13726 C0SBR8 3025935 EC50 = 2800 nM T13726 CK6X4W 3025936 EC50 = 2300 nM T13726 CK3N2G 3035780 EC50 = 86 nM T13726 CUL8F1 5354022 EC50 = 2700 nM T13726 CGL71X 6366726 EC50 = 11 nM T13726 C5EON6 6366727 EC50 = 592 nM T13726 C62YGF 6366732 EC50 > 0.001 nM T13726 CK4UA6 6366733 EC50 = 112 nM T13726 CLF4M5 6366734 EC50 = 105 nM T13726 CA5GS8 6438168 EC50 = 201 nM T13726 C7C9SR 6439768 EC50 > 10000 nM T13726 C16ZSG 6439929 IC50 = 33000 nM T13726 CGTB79 6440940 EC50 = 27000 nM T13726 C5LH2R 6441236 EC50 = 10000 nM T13726 CJHW10 6441985 EC50 = 385 nM T13726 CHA3C2 6447986 EC50 = 2700 nM T13726 C3F4GD 6447987 EC50 = 2800 nM T13726 CVIT54 6491146 EC50 = 27000 nM T13726 CZ2N9P 7023630 EC50 = 27000 nM T13726 CG4FM8 7745122 EC50 = 160 nM T13726 CRXY80 7745146 EC50 = 280 nM T13726 C9SX8K 7745148 EC50 = 5000 nM T13726 CBE62R 9799320 EC50 = 130 nM T13726 CRK31P 9799442 EC50 = 52 nM T13726 COP9S7 9799477 EC50 = 4 nM T13726 CSNI93 9799841 EC50 = 207 nM T13726 CJ3ZM0 9801665 Ki = 3 nM T13726 CX2HY4 9801929 EC50 = 332 nM T13726 CY1V5S 9802575 EC50 = 540 nM T13726 C8P4UD 9803186 Ki = 4.8 nM T13726 CW7D0R 9810431 Ki = 138 nM T13726 CBV6Y2 9818688 EC50 = 2500 nM T13726 CUJ14W 9819890 EC50 > 10000 nM T13726 CEK1O4 9820039 EC50 = 210 nM T13726 C1A2UO 9820391 EC50 = 26 nM T13726 CQI49S 9820393 EC50 = 115 nM T13726 CIN7X1 9820545 EC50 = 31 nM T13726 CPMX25 9820546 EC50 = 34 nM T13726 C4WK5D 9824444 IC50 = 8 nM T13726 C26HXU 9842010 EC50 = 51 nM T13726 C94MFP 9842758 EC50 = 3 nM T13726 CQFA96 9845057 Ki = 1.5 nM T13726 CQ1ZH6 9847065 IC50 = 4 nM T13726 C3X8NU 9858424 IC50 >= 100000 nM T13726 CWOG69 9864474 EC50 = 300 nM T13726 CB3NF2 9866384 EC50 = 3.3 nM T13726 CJ08SK 9867780 EC50 = 3.4 nM T13726 CAE0R3 9868664 Ki = 4.1 nM T13726 CF12VS 9869030 IC50 = 430 nM T13726 CRC51S 9869157 IC50 = 13.7 nM T13726 CXAE08 9884280 EC50 = 1000 nM T13726 CA0TS6 9884959 EC50 = 30 nM T13726 CSK5B8 9885521 EC50 > 1000 nM T13726 C6ZR5D 9885730 Ki = 1 nM T13726 C3CS9R 9886082 EC50 = 381 nM T13726 C5AD1H 9886137 EC50 = 5 nM T13726 CKNQ14 9887034 EC50 = 74 nM T13726 CG3JR4 9887949 EC50 = 51 nM T13726 C90UXQ 9889347 EC50 = 6.8 nM T13726 C8MK1Y 9889522 Ki = 900 nM T13726 CS3AR1 9904203 EC50 = 820 nM T13726 C2WFX1 9905729 Ki = 150 nM T13726 C2D9WJ 9906413 EC50 = 455 nM T13726 CRS67U 9906421 EC50 = 470 nM T13726 C9AJZ7 9906514 EC50 = 13 nM T13726 C7E0IO 9907433 EC50 = 294 nM T13726 CL1K7B 9907909 EC50 = 63 nM T13726 COS0D4 9908099 Ki = 4 nM T13726 CSF7G1 9908857 Ki = 14 nM T13726 C0A3UZ 9911319 Ki = 0.8 nM T13726 CSW2Y8 9929026 Ki = 20 nM T13726 CQ6I7G 9946524 Ki > 3000 nM T13726 CIS1Z0 9948900 EC50 > 10000 nM T13726 C9VEF0 9949645 EC50 = 2971 nM T13726 C6CI3S 9950957 EC50 = 514 nM T13726 C0GLF2 9952045 EC50 = 6.4 nM T13726 CDZC95 9952534 EC50 = 750 nM T13726 C6JLI1 9973307 EC50 = 1200 nM T13726 CVM8I3 9973559 EC50 = 4700 nM T13726 CV1A3K 9974457 EC50 > 1000 nM T13726 C63OUJ 9976842 EC50 > 1000 nM T13726 CAE52Z 9997909 EC50 = 2500 nM T13726 C7VS6O 9998151 EC50 = 380 nM T13726 C05EXS 9998870 EC50 = 83 nM T13726 CL7X4Y 9999621 EC50 > 10000 nM T13726 CM1BQ5 10003577 Ki = 2.3 nM T13726 C7ER2L 10020788 EC50 > 10000 nM T13726 CBR3O2 10021705 EC50 = 650 nM T13726 CZP71W 10022432 EC50 = 2220 nM T13726 CN6LP5 10022568 EC50 > 10000 nM T13726 C8RSG9 10043365 EC50 = 55 nM T13726 CC0N1S 10043729 EC50 = 330 nM T13726 CE60FI 10065757 Ki = 3 nM T13726 C2C0GJ 10066739 EC50 = 2400 nM T13726 CFQ1Y3 10073992 Ki = 3 nM T13726 C4VU6T 10087372 EC50 = 2400 nM T13726 CXL0Y3 10089642 EC50 = 2200 nM T13726 CC8R9M 10093918 Ki = 3800 nM T13726 CZI69W 10112018 Ki = 69.2 nM T13726 CPX6Q5 10115123 Ki = 394.7 nM T13726 CCKL65 10135144 EC50 = 29 nM T13726 CD3B1K 10135277 EC50 = 20 nM T13726 C59GXP 10135960 EC50 = 6 nM T13726 CO4S6H 10137005 EC50 = 86 nM T13726 CQYW32 10137940 Ki = 14 nM T13726 CU2H3N 10156587 EC50 = 42 nM T13726 C2S1QO 10158313 Ki = 648 nM T13726 C6KS9R 10202323 Ki = 44 nM T13726 CP96OH 10204841 IC50 = 22 nM T13726 CTKY45 10206438 Ki = 12 nM T13726 C90YNI 10207221 Ki = 7 nM T13726 C1O4PN 10207439 Ki = 3 nM T13726 C0DS6Q 10223041 Ki = 2078.3 nM T13726 C6N5OK 10224145 EC50 = 1442 nM T13726 CZM6O3 10225147 Ki = 47 nM T13726 C7L4CJ 10225689 Ki = 740 nM T13726 CKR51I 10225690 Ki = 1.6 nM T13726 C0AV2Z 10226478 Ki = 198 nM T13726 CUV8S0 10249942 IC50 = 1 nM T13726 CZY92F 10271982 Ki = 131 nM T13726 C1K8YO 10272875 Ki = 20 nM T13726 COD29A 10272879 Ki = 29.6 nM T13726 CH5G4X 10273806 Ki = 271 nM T13726 C0WRE7 10273807 Ki = 6 nM T13726 C2P8CN 10274512 Ki = 7.4 nM T13726 CIKB68 10274731 EC50 = 40 nM T13726 C1LN6I 10274852 EC50 = 38 nM T13726 CCD7A5 10276434 Ki = 3.2 nM T13726 C54TLG 10286680 IC50 >= 100000 nM T13726 CP3MN0 10289172 EC50 = 0.9 nM T13726 C1LUP9 10294771 Ki = 22 nM T13726 C6FT2B 10294841 Ki = 6 nM T13726 C2N9DJ 10296557 EC50 = 3976.3 nM T13726 C27ZPC 10297135 Ki = 161 nM T13726 CS6N3M 10298831 Ki = 1.6 nM T13726 CY1J5M 10308975 Ki = 4 nM T13726 C61TSO 10314077 EC50 = 2500 nM T13726 CUZR60 10314977 EC50 = 300 nM T13726 CVQ7Z6 10316839 EC50 = 2019 nM T13726 C6C5GP 10320109 Ki = 1800 nM T13726 CO5Q7F 10338255 EC50 = 11300 nM T13726 C5LV9X 10358286 EC50 = 2600 nM T13726 CK0S3U 10360455 EC50 = 6 nM T13726 C2XBM9 10362613 EC50 = 21 nM T13726 CUEF37 10362997 EC50 = 300 nM T13726 CG01ED 10383375 EC50 = 197 nM T13726 CZTK13 10405638 EC50 = 3100 nM T13726 CA6FH2 10427143 EC50 = 460 nM T13726 C4TBM8 10449810 EC50 = 2900 nM T13726 CXQ9S4 10450790 EC50 = 1820 nM T13726 CXA0N9 10458226 Ki = 3800 nM T13726 C8TK9E 10473090 EC50 > 10000 nM T13726 C0CHL5 10474101 EC50 = 200 nM T13726 CL31KB 10499086 EC50 = 253 nM T13726 CF87BZ 10523774 EC50 = 384 nM T13726 C2TP9D 10598286 Ki = 484 nM T13726 CS96IV 10619935 Ki = 4 nM T13726 C4TO6H 10620598 EC50 = 5 nM T13726 CE1OC7 10644298 Ki = 620 nM T13726 CH3D5N 10645862 Ki > 1000 nM T13726 CVQ6L1 10759115 EC50 = 3100 nM T13726 CMXI39 10804037 EC50 = 2800 nM T13726 CJ57NB 10916642 Ki = 2 nM T13726 C8UG3F 10926235 EC50 = 4 nM T13726 CURV10 10926384 EC50 = 2 nM T13726 CWM7E2 10936808 Ki = 1 nM T13726 CTB3E6 10937639 Ki = 1 nM T13726 CF7DZ3 10938844 IC50 = 13 nM T13726 CG48CT 11025742 Ki = 2 nM T13726 C6F1MJ 11079184 Ki = 3 nM T13726 CO50RB 11080831 IC50 = 16 nM T13726 C5R1KA 11178007 IC50 = 10 nM T13726 CIO2Y3 11220435 EC50 = 8660 nM T13726 C34EXF 11221031 Ki > 1000 nM T13726 CUP91B 11234875 EC50 = 97 nM T13726 CF12QM 11256032 EC50 = 9600 nM T13726 CTX20E 11258568 IC50 = 500 nM T13726 CFMR40 11327597 IC50 = 6 nM T13726 CF6XT3 11349910 EC50 = 22 nM T13726 C5F6NY 11370831 EC50 = 15900 nM T13726 C3FQ4D 11416475 Ki = 138 nM T13726 CC5M6P 11416879 EC50 = 106 nM T13726 CA4PZ9 11430044 IC50 = 120 nM T13726 CW9VO2 11441858 IC50 = 270 nM T13726 C4BW0C 11461003 EC50 = 30 nM T13726 CIHX19 11559459 EC50 = 19 nM T13726 C6ZI9M 11617486 EC50 = 215 nM T13726 C7KQZ1 11725331 EC50 = 300 nM T13726 C9YU4D 11725332 EC50 = 55 nM T13726 CY85CP 11749701 EC50 = 10 nM T13726 CC40ME 11793226 EC50 = 46 nM T13726 C0WA5F 11793407 Ki = 2 nM T13726 C4QYX8 11962184 Ki = 8 nM T13726 C38KZG 11978565 EC50 = 27000 nM T13726 C1AOP8 11978570 EC50 = 13000 nM T13726 C7UWV3 12112296 EC50 = 298 nM T13726 CIQJ20 12112298 EC50 = 275 nM T13726 CQ9YE5 12358678 EC50 = 13 nM T13726 C4U3BH 12358681 EC50 = 4 nM T13726 CY5AZ1 13187576 EC50 > 6400 nM T13726 C5TS1Q 13413729 EC50 = 2800 nM T13726 CT41DZ 14557465 EC50 = 1100 nM T13726 CNS9T8 15434197 Ki = 5 nM T13726 C8Z7RF 16041073 EC50 = 1.8 nM T13726 C62ZGE 16041074 EC50 = 61.2 nM T13726 C12UOE 16041242 EC50 = 96.6 nM T13726 C84SDA 16128741 EC50 = 173.1 nM T13726 CRB7Z6 16128818 EC50 = 19.2 nM T13726 C06CRH 16128819 EC50 = 16.3 nM T13726 C4Z2HV 16128820 EC50 = 7.2 nM T13726 CDT6P8 16128821 EC50 = 18.3 nM T13726 C7O4UQ 16128822 EC50 = 45.9 nM T13726 CRL06N 16128823 EC50 = 3.4 nM T13726 CV8TP1 16221202 EC50 = 12200 nM T13726 CT32AS 16221263 EC50 = 16400 nM T13726 CQL8O3 16222898 EC50 = 1600 nM T13726 CJ74NB 16794302 EC50 > 30000 nM T13726 CD1P2E 17753147 EC50 = 67.3 nM T13726 CU3BR6 17755855 EC50 = 4840 nM T13726 C3P6XD 19002087 EC50 = 89 nM T13726 CVA8T2 20117108 IC50 = 11000 nM T13726 CY7P2M 20707149 EC50 = 350 nM T13726 CV1C4A 22226112 EC50 > 1000 nM T13726 C41JDY 22400850 EC50 > 30000 nM T13726 CA59NU 22686157 EC50 > 30000 nM T13726 C0M9JB 22688013 EC50 = 13000 nM T13726 CP2CA5 23005221 EC50 = 80 nM T13726 CSX90U 23626229 IC50 = 500 nM T13726 C5JSU9 23626230 IC50 = 95 nM T13726 CAF52J 23626231 IC50 = 190 nM T13726 CTE1N2 24748569 EC50 > 10000 nM T13726 C15NSJ 24828803 EC50 = 7300 nM T13726 CO31MA 24828805 EC50 = 6100 nM T13726 CW51RK 24828806 EC50 = 1500 nM T13726 CS05HD 24857921 EC50 = 66 nM T13726 CL0K5P 25006094 EC50 = 19 nM T13726 C3A2LN 25006098 EC50 = 450 nM T13726 C9N4PO 25195030 IC50 = 4100 nM T13726 CQUB90 25195031 IC50 = 3200 nM T13726 C0A2XU 29288275 EC50 = 1100 nM T13726 CT4J7Z 41500207 IC50 = 7000 nM T13726 C1SXJ3 44274894 IC50 = 21 nM T13726 CS7U6L 44285287 EC50 = 1500 nM T13726 CPA87R 44287651 Ki = 5 nM T13726 C1K8FB 44287715 IC50 = 11 nM T13726 CI83JY 44287875 Ki = 7 nM T13726 CB8PI2 44304045 EC50 = 4 nM T13726 CIVH74 44316525 Ki = 66 nM T13726 CAP68W 44316543 Ki = 4 nM T13726 CAI2Z5 44316544 Ki = 4 nM T13726 C0YQ8H 44316756 Ki = 15 nM T13726 C6Q1CA 44316796 Ki = 3 nM T13726 CLK5H0 44316811 Ki = 38 nM T13726 CK48CT 44321880 EC50 = 2800 nM T13726 CXV0B4 44321951 EC50 = 2800 nM T13726 CH8T3V 44325132 EC50 = 59 nM T13726 C1KUN0 44325759 EC50 = 51 nM T13726 CLB6X7 44325767 Ki > 1000 nM T13726 C39LIO 44325862 Ki = 2.7 nM T13726 CK6JC0 44338117 Ki = 8.2 nM T13726 CP51SQ 44338305 EC50 = 805.8 nM T13726 CG6H2T 44353335 Ki = 3 nM T13726 CW0T6K 44353336 Ki = 0.8 nM T13726 C8K0AB 44353347 Ki = 4.4 nM T13726 C3DYE9 44353422 Ki = 1 nM T13726 C5DTY3 44353441 Ki = 2.6 nM T13726 C2M8TN 44353456 IC50 = 10.7 nM T13726 CVKA40 44353466 Ki = 6.1 nM T13726 C8J5SA 44353480 IC50 = 5.1 nM T13726 CIB15X 44353481 IC50 = 5.3 nM T13726 CY9XP2 44366042 EC50 > 10000 nM T13726 CWC73Q 44375294 IC50 >= 100000 nM T13726 C1AM4Y 44377164 EC50 = 713 nM T13726 C05RAC 44377446 Ki = 11 nM T13726 CPW0M2 44377447 Ki = 21 nM T13726 CDU3F0 44410404 Ki = 18 nM T13726 CRW3F9 44410405 Ki = 257 nM T13726 CJX92G 44410453 Ki = 21 nM T13726 C1YKC7 44410518 Ki = 103 nM T13726 CI64YQ 44410534 Ki = 644 nM T13726 CE6W1Y 44410535 Ki = 529 nM T13726 CCS4X0 44410540 Ki = 37 nM T13726 CQVY89 44410541 Ki = 31 nM T13726 CLR9U4 44410562 Ki = 122 nM T13726 CXI98E 44410565 Ki = 21 nM T13726 C0ZIF2 44410568 Ki = 67 nM T13726 CW4YU7 44410575 Ki = 17 nM T13726 CV0TB9 44410576 Ki = 121 nM T13726 C9L6TA 44410610 Ki = 63 nM T13726 CKY50J 44410620 Ki = 42 nM T13726 CO2AF5 44410623 Ki = 47 nM T13726 C2R7KB 44410653 Ki = 254 nM T13726 C2QW1R 44410654 Ki = 103 nM T13726 C6D2SZ 44427044 IC50 = 2000 nM T13726 CN62HA 44427046 IC50 = 1600 nM T13726 CMP2K5 44427047 IC50 = 1000 nM T13726 C8DGP5 44427048 IC50 = 670 nM T13726 CB9J8M 44427049 IC50 = 4900 nM T13726 C9PL1O 44427050 IC50 = 1400 nM T13726 C81PRC 44427051 IC50 = 450 nM T13726 C2PRD4 44427052 IC50 = 360 nM T13726 C8UIF4 44427053 IC50 = 130 nM T13726 C8ZSP3 44427055 IC50 = 420 nM T13726 CW1E9H 44427056 IC50 = 780 nM T13726 CXUN75 44427057 IC50 = 1300 nM T13726 C28ACU 44427058 IC50 = 2000 nM T13726 C1T5WL 44427059 IC50 = 190 nM T13726 COZ5M2 44427061 IC50 = 460 nM T13726 C3AM2J 44427063 IC50 = 450 nM T13726 C8ATQ5 44427065 IC50 = 450 nM T13726 CKO3F2 44427067 IC50 = 1000 nM T13726 CX3OG7 44427068 IC50 = 3900 nM T13726 CZ7HY4 44427070 IC50 = 11000 nM T13726 CRI4K1 44427073 IC50 = 890 nM T13726 C8F0OR 44427074 IC50 = 970 nM T13726 CUK4H1 44427075 IC50 = 4600 nM T13726 C2TV8F 44427076 IC50 = 1100 nM T13726 C2Q8TM 44427077 IC50 = 3000 nM T13726 CTW0J5 44427078 IC50 = 320 nM T13726 CFD81J 44427079 IC50 = 2100 nM T13726 CC4DG9 44427080 IC50 = 520 nM T13726 CP28DC 44427081 IC50 = 530 nM T13726 CTGI62 44433353 IC50 > 100000 nM T13726 CTLZ45 44433354 IC50 > 100000 nM T13726 CB9T1J 44433355 IC50 > 10000 nM T13726 CZX0Q3 44433356 IC50 = 7100 nM T13726 C7HLK1 44433357 IC50 = 1800 nM T13726 CXRT02 44433364 IC50 = 5600 nM T13726 CHR04N 44433371 IC50 = 4500 nM T13726 CL3P5H 44433377 IC50 = 2900 nM T13726 C4ZM3P 44433390 IC50 = 900 nM T13726 CG2DT7 44433396 IC50 = 1700 nM T13726 C8ILT2 44433397 IC50 = 4100 nM T13726 C6SJ9X 44433398 IC50 = 2500 nM T13726 CAPL02 44433403 IC50 = 880 nM T13726 CA9VR6 44433404 IC50 = 720 nM T13726 C2OK4E 44433405 IC50 = 3100 nM T13726 CEJ0N7 44433408 IC50 = 3800 nM T13726 C18NUW 44433410 IC50 = 14000 nM T13726 CH1ET8 44433412 IC50 = 7300 nM T13726 CYNW40 44433414 IC50 = 5200 nM T13726 CW7A2C 44433415 IC50 = 3400 nM T13726 CS3Y9P 44433416 IC50 = 2800 nM T13726 CTX35K 44433437 IC50 = 2400 nM T13726 CNJC69 44433438 IC50 = 840 nM T13726 CCZP28 44433440 IC50 = 250 nM T13726 C4ZC3E 44433443 IC50 = 370 nM T13726 C7QX4Y 44433447 IC50 = 340 nM T13726 CAY4N0 44433449 IC50 = 550 nM T13726 C7DAP4 44433451 IC50 = 200 nM T13726 CZE62U 44433452 IC50 = 850 nM T13726 CUWH91 44433453 IC50 = 5200 nM T13726 CVP4Y8 44433454 IC50 = 400 nM T13726 C9UHL7 44433456 IC50 = 510 nM T13726 CXH9P3 44433457 IC50 = 4400 nM T13726 CPSO05 44433458 IC50 = 1200 nM T13726 CXK5F6 44433460 IC50 = 190 nM T13726 C7S4ZD 44433463 IC50 = 220 nM T13726 CQV0D2 44433465 IC50 = 130 nM T13726 C8YL2K 44433466 IC50 = 430 nM T13726 CB42MF 44433467 IC50 = 470 nM T13726 CI8RE2 44433468 IC50 = 1400 nM T13726 C6F4YV 44433469 IC50 = 1500 nM T13726 CO4S8D 44433470 IC50 = 1100 nM T13726 C0V7CP 44433474 IC50 = 1200 nM T13726 CJN69Z 44433476 IC50 = 3400 nM T13726 CLFW81 44433477 IC50 = 1300 nM T13726 CR0N1W 44442494 EC50 = 39.1 nM T13726 CZL4P9 44442496 EC50 > 10000 nM T13726 C4HUT2 44442497 EC50 = 27.9 nM T13726 CU85RK 44442498 EC50 = 527 nM T13726 CA2H8W 44442502 EC50 = 760 nM T13726 C4TK6U 44442504 EC50 = 37.7 nM T13726 C8CH2K 44442512 EC50 = 1.4 nM T13726 CA50DX 44442514 EC50 = 70.2 nM T13726 CDYR68 44442515 EC50 = 36.5 nM T13726 C4JCR8 44442516 EC50 = 361 nM T13726 CMWX53 44442517 EC50 = 115.8 nM T13726 CWM9G1 44442518 EC50 = 5 nM T13726 C27FTL 44442519 EC50 = 207.5 nM T13726 CT09ZO 44442520 EC50 = 144 nM T13726 C4JSO9 44442521 EC50 = 2.3 nM T13726 C58GAP 44442522 EC50 = 361 nM T13726 CNU82F 44442523 EC50 = 10 nM T13726 CE47QM 44442524 EC50 = 198 nM T13726 CFG4B7 44442602 EC50 > 10000 nM T13726 CT24UG 44442603 EC50 = 1200 nM T13726 CWY23H 44442608 EC50 = 24.3 nM T13726 CC2G5I 44442609 EC50 = 2.1 nM T13726 CFQ59C 44442610 EC50 = 1.8 nM T13726 CRI0J3 44460654 Ki > 2200 nM T13726 CR5SI0 44476535 EC50 > 10000 nM T13726 CEA20Z 44571531 IC50 > 10000 nM T13726 CG02HN 44571532 IC50 > 10000 nM T13726 CDZ84V 44571568 IC50 = 5200 nM T13726 CF21WB 44571569 IC50 = 2700 nM T13726 CA9FT0 44571643 IC50 > 10000 nM T13726 CK36AF 45483161 Ki = 81 nM T13726 C9KWZ7 45483162 Ki = 161 nM T13726 C3UX8H 45483163 Ki = 12 nM T13726 CCA3G0 46224594 IC50 = 2400 nM T13726 CBH2U9 46835962 EC50 = 367 nM T13726 CEA7F3 46893394 EC50 = 820 nM T13726 CN9L7G 46916268 EC50 > 15000 nM T13726 C42EMT 46933534 EC50 = 205 nM T13726 C6M3FK 46933689 EC50 = 3.8 nM T13726 CUD91T 49862248 EC50 > 10000 nM T13726 C1DNC5 49865443 EC50 = 1000 nM T13726 CV17PS 49865445 EC50 = 1000 nM T13726 CQWG01 49865446 EC50 = 1000 nM T13726 C6F7SH 49870954 EC50 = 290 nM T13726 CHE75O 49870965 EC50 = 160 nM T13726 CCQN30 49870966 EC50 = 160 nM T13726 CO74VZ 53218383 EC50 = 25400 nM T13726 C08ADT 53318572 EC50 = 280 nM T13726 C50FJA 53319895 EC50 = 110 nM T13726 CEGB39 53319896 EC50 = 160 nM T13726 C52JRP 53322528 EC50 = 180 nM T13726 CT4JC1 53323864 EC50 = 330 nM T13726 C4CP2D 53325142 EC50 = 160 nM T13726 CQV3T7 53355501 EC50 = 9220 nM T13726 CZ45ND 54588772 IC50 = 1600 nM T13726 CW4GB2 54588773 IC50 = 6290 nM T13726 C5EZ4U 54588774 IC50 = 3150 nM T13726 CUDH10 54588775 IC50 = 10650 nM T13726 CUH9M4 54588776 IC50 >= 100000 nM T13726 C4F2QC 54588811 IC50 >= 100000 nM T13726 C1NO4X 54588812 IC50 >= 100000 nM T13726 CUJ31A 54588813 IC50 = 4730 nM T13726 CWM49I 54588814 IC50 = 8270 nM T13726 CXL6G9 54588815 IC50 >= 100000 nM T13726 CG58EP 54588816 IC50 >= 100000 nM T13726 C83JOA 54588850 IC50 >= 100000 nM T13726 C09YKD 54588851 IC50 >= 100000 nM T13726 C0O2MI 54588852 IC50 >= 100000 nM T13726 C6YZO4 54588856 IC50 >= 100000 nM T13726 CPSO83 54588890 IC50 >= 100000 nM T13726 C8FR2C 54588891 IC50 >= 100000 nM T13726 CYPU61 54588892 IC50 = 3080 nM T13726 CWBY91 54588893 IC50 >= 100000 nM T13726 C5Y3FP 54588894 IC50 >= 100000 nM T13726 CAFZ93 54589361 IC50 >= 100000 nM T13726 CZ3E9U 54589362 IC50 = 10000 nM T13726 C5EW6P 54589363 IC50 >= 100000 nM T13726 CMS60L 54589364 IC50 = 5710 nM T13726 C5ZX4B 54597874 EC50 > 10000 nM T13726 CB84WZ 59205486 EC50 = 18000 nM T13726 C6ER1K 59444433 EC50 = 720 nM T13726 CZK03B 59444434 EC50 = 100 nM T13726 C1ENS2 59444436 EC50 = 620 nM T13726 CIO69D 59853119 EC50 = 14300 nM T13726 C6AZ0X 60148508 EC50 = 3370 nM T13726 CO4P2S 60148514 EC50 = 4220 nM T13726 CN20JG 60148515 EC50 = 9960 nM T13726 C42FDY 60163732 EC50 = 19.5 nM T13726 CH95XR 60165808 EC50 > 34700 nM T13726 CABW49 60166111 EC50 = 20910 nM T13726 CNR48W 62216411 EC50 > 30000 nM T13726 C9S5EN 64222254 EC50 > 30000 nM T13726 CX1P8I 67042254 IC50 > 10000 nM T13726 CGL2E4 70868689 EC50 = 3400 nM T13726 C27OVL 71461789 EC50 = 143 nM T13726 C3ARJ0 71544866 EC50 > 20700 nM T13726 CYL3F6 71546517 EC50 > 44500 nM T13726 C7VJN5 71547126 EC50 = 8400 nM T13726 C9K7YI 71584530 EC50 = 83 nM T13726 CHU9X0 71584534 EC50 = 633 nM T13726 CD3GZ8 71584654 EC50 = 155 nM T13726 C46HSQ 71584655 EC50 = 15 nM T13726 CUT25I 71601083 EC50 = 19460 nM T13726 C03QGP 71601234 EC50 = 18440 nM T13726 CB0U7G 71601367 EC50 = 10720 nM T13726 CU70LB 71601660 EC50 = 7000 nM T13726 CO67YL 71601664 EC50 = 10010 nM T13726 CCX30R 71717207 Ki > 2200 nM T13726 C9G2SH 73054430 EC50 = 120 nM T13726 CTZ3K4 73296637 EC50 = 770 nM T13726 CVW1H0 73350281 Ki = 19 nM T13726 CX65SN 73659166 IC50 = 10000 nM T13726 C7OA9K 73775427 EC50 = 169 nM T13726 CY7SE1 76317515 IC50 > 25000 nM T13726 CBG04C 80198302 EC50 = 10600 nM T13726 C3PI7Z 82483008 EC50 = 4300 nM T13726 C5V8NG 90644073 EC50 = 160 nM T13726 CYQ9N5 101905252 EC50 = 780 nM T13726 C8CJR5 102004339 EC50 > 100000 nM T13726 CW27MY 118063735 EC50 > 10000 nM T13726 CSX68I 118736632 EC50 = 12 nM T13726 CF1H7K 118736686 EC50 = 450 nM T13726 CFUC59 118796352 EC50 = 6.31 nM T13726 C6TBD2 121345502 EC50 > 20000 nM T13726 CAN4E2 122191999 EC50 = 50 nM T13726 CFG36H 122192000 EC50 = 23 nM T13726 CU0XD9 122192001 EC50 = 22 nM T13726 C1QVY6 122192002 EC50 = 80 nM T13726 C58HKI 127030410 EC50 = 1000 nM T13726 CFBD60 127033242 EC50 = 50.12 nM T13726 CPJ37K 127033515 EC50 = 25.12 nM T13726 CR74DS 127033518 EC50 = 50.12 nM T13726 CZR8F2 127033519 EC50 = 125.89 nM T13726 C0L4ZF 127033523 EC50 = 15.85 nM T13726 C8Q0JO 131750108 EC50 = 22 nM T13726 C38PLT 135588490 IC50 = 2450 nM T13726 CSQ30M 136211075 IC50 = 2810 nM T13726 C2WG9L 138393074 EC50 = 970 nM T13726 C2OJ9E 141259219 EC50 = 11800 nM T13726 C7N6KH 145950441 EC50 = 23600 nM T13726 CRTB69 145952096 EC50 = 9100 nM T13726 CLND09 145957286 EC50 = 24000 nM T13726 CO5LP2 145959006 EC50 = 8000 nM T13726 CCF02H 145964530 IC50 = 4400 nM T13726 C56SHA 145964597 IC50 = 4600 nM T13726 C5H8EZ 145965425 IC50 = 2000 nM T13726 C98CHS 145977976 IC50 = 11100 nM T13726 CM8T6X 145982686 EC50 = 19000 nM T13726 C1QZ7W 145986715 IC50 = 2000 nM T13726 C7X3AL 153763221 EC50 = 9600 nM T13726 CUNF95 155513665 EC50 = 19800 nM T13726 C3Z6VL 155514089 EC50 = 6800 nM T13726 CGO6X4 155515480 EC50 = 6000 nM T13726 CWR01U 155517898 EC50 > 30000 nM T13726 C7DN5A 155520617 EC50 > 30000 nM T13726 CT4HM2 155524204 EC50 = 3500 nM T13726 C95KYP 155526365 EC50 = 2100 nM T13726 COG5A0 155530735 EC50 = 9800 nM T13726 C2QTX3 155530866 EC50 = 1500 nM T13726 C4JD0I 155531001 EC50 = 10000 nM T13726 CPXG96 155531076 EC50 = 27 nM T13726 CE7I8Q 155534885 EC50 = 36400 nM T13726 CX2JR0 155535627 EC50 = 3700 nM T13726 CE7OD6 155538138 EC50 = 210 nM T13726 C1TMV9 155539075 EC50 = 1100 nM T13726 CEM97Q 155539095 EC50 = 6700 nM T13726 COP7X8 155539171 IC50 > 10000 nM T13726 C3R9YL 155539254 EC50 = 25000 nM T13726 C7E9KD 155539294 EC50 = 4200 nM T13726 CR9Y8W 155541027 EC50 = 9100 nM T13726 CP3I4H 155541634 EC50 = 950 nM T13726 C2QGR5 155549327 EC50 = 10000 nM T13726 C6GQJ9 155552325 EC50 = 275 nM T13726 C80ZVT 155556139 EC50 > 30000 nM T13726 CJQ54R 155556924 EC50 = 30200 nM T13726 CIO4S2 155557691 EC50 = 93 nM T13726 CM52UW 155560868 EC50 = 1400 nM T13726 CG3D8J 155564760 EC50 = 470 nM T13726 CX7OR2 155566024 EC50 = 8000 nM T13726 C2A1UC 10429766 Ki = 3 nM T13726 D02YHD 11755040 IC50 = 900 nM T13726 D04DQJ 72303 EC50 = 11800 nM T13726 D09XCX 5694 EC50 = 9100 nM T13726 D0G6JM 5289501 EC50 > 0.001 nM T13726 D0Q9FZ 6442223 EC50 = 2 nM T94324 D00SQN 12136798 IC50 = 235 nM T94324 D0E3SH 6918837 Ki = 5.1 nM T94324 D0E7PQ 5311 Ki = 40 nM T94324 D0L7LC 5352062 IC50 = 11 nM T94324 D05KED 53340666 IC50 = 125.89 nM T94324 D07FPY 6918877 Ki = 18.9 nM T94324 D09XIZ 11538455 Ki = 0.05 nM T94324 D0B3FV 6445533 IC50 = 8.41 nM T94324 D0E6UZ 54575456 IC50 = 2.8 nM T94324 D0L2UQ 49855250 Ki = 23 nM T94324 D0M8FD 4261 IC50 = 11100 nM T94324 D0V0SL 11749858 IC50 = 3.981 nM T94324 D0XT6W 6918638 Ki = 59 nM T94324 D0Z4RC 24756910 IC50 = 26.1 nM T94324 D0J8OC 5186 IC50 = 300 nM T94324 D00HXJ 118884610 Ki = 452 nM T94324 D0N2DK 72710871 IC50 = 10.6 nM T94324 D0QX3G 71532921 IC50 = 79.43 nM T94324 C18ENP 6918846 Ki = 23 nM T94324 CJ07ZA 9800555 IC50 = 78 nM T94324 CC0EU7 9828788 IC50 = 3.9 nM T94324 C7RC1E 10309899 IC50 = 4.3 nM T94324 C8G5WP 11210533 IC50 = 8100 nM T94324 C0TPN8 11254230 IC50 = 280 nM T94324 CI7W3O 11267278 IC50 = 1540 nM T94324 CM6ZW2 11279156 IC50 = 3430 nM T94324 C2F9NT 11558827 IC50 = 176 nM T94324 CG9OC4 11682502 IC50 = 42.6 nM T94324 CYB26W 11688197 IC50 = 899 nM T94324 CC3R6T 11777910 IC50 = 50 nM T94324 CE4Z0Y 11844891 IC50 = 5210 nM T94324 C9G1BN 11993595 IC50 = 4700 nM T94324 CH5JS7 11993694 IC50 = 240 nM T94324 C06UTF 13507024 IC50 = 40 nM T94324 C2D1KP 15983982 Ki = 13 nM T94324 CHB82E 15986417 IC50 > 100000 nM T94324 C52EVH 15986418 IC50 = 11000 nM T94324 CS1QO9 15986509 IC50 = 91000 nM T94324 CFK8J5 16068056 Ki = 34 nM T94324 CMQP70 16068495 Ki = 34 nM T94324 CT84XO 16068594 Ki = 29 nM T94324 CF3ZG5 16068595 Ki = 28 nM T94324 CL60CA 16068912 Ki = 19 nM T94324 CUG50I 16733294 IC50 = 46.1 nM T94324 CWO7V0 16733295 IC50 = 173 nM T94324 C4W0PG 16733410 IC50 = 28.3 nM T94324 C0MO3Z 16733411 IC50 = 11.1 nM T94324 C3QL4X 16733412 IC50 = 29700 nM T94324 CV54SY 16733414 IC50 = 10700 nM T94324 C1VCX2 16733415 IC50 = 178 nM T94324 CXN07K 16733416 IC50 > 30000 nM T94324 CP9AR8 16733417 IC50 = 42.1 nM T94324 CUE62T 16733590 IC50 = 8780 nM T94324 C17GDO 24779722 IC50 = 179 nM T94324 CLT5J2 24881257 IC50 = 188 nM T94324 C5GCM1 24881328 IC50 = 112 nM T94324 C8QVB1 24881329 IC50 = 86.5 nM T94324 CU0AM3 24881330 IC50 = 18.5 nM T94324 CQM51L 24881331 IC50 = 27.7 nM T94324 C4KH8F 24881332 IC50 = 64.7 nM T94324 C1KA3V 24881333 IC50 = 74.8 nM T94324 C47APB 24881402 IC50 = 19.2 nM T94324 CSN8W1 24881403 IC50 = 24.5 nM T94324 C1UQ3K 24881404 IC50 = 36.1 nM T94324 C51TMH 24881405 IC50 = 34.3 nM T94324 C9EZI7 24881406 IC50 = 13 nM T94324 C6P3HS 24881407 IC50 = 70.1 nM T94324 CZ3TU1 24881464 IC50 = 55.7 nM T94324 CDI49N 24881465 IC50 = 17.6 nM T94324 CQGP87 24881466 IC50 = 15.8 nM T94324 CC0R9O 24938735 IC50 = 0.5 nM T94324 CF03HD 24948905 IC50 = 690 nM T94324 CHP8O6 24948906 IC50 = 17.5 nM T94324 C1KRT8 24948907 IC50 = 840 nM T94324 CKY2P8 24948908 IC50 = 44.9 nM T94324 C25CFI 24948909 IC50 = 401 nM T94324 CWQ04Z 24948910 IC50 = 73 nM T94324 CM9I3X 24951310 IC50 = 155 nM T94324 CX1YF8 24951311 IC50 = 852 nM T94324 CV10XU 24951312 IC50 = 28.2 nM T94324 CD6KV0 24951313 IC50 = 891 nM T94324 CQY9Z0 24951314 IC50 = 90.7 nM T94324 CX69SY 25066355 IC50 = 1530 nM T94324 CF8VP4 25066356 IC50 = 683 nM T94324 CS9XH7 25066547 IC50 = 958 nM T94324 C46AGN 25066548 IC50 = 70.7 nM T94324 CJF2M7 25066549 IC50 = 320 nM T94324 CCD5M7 25227504 IC50 = 62.5 nM T94324 CK0D5S 25227505 IC50 = 152 nM T94324 CN97JP 25227508 IC50 = 190 nM T94324 CW8R1B 25227513 IC50 = 200 nM T94324 C43BHY 25269097 IC50 = 42 nM T94324 CJ1RQ7 42598706 IC50 = 1350 nM T94324 CDT65Y 42631047 IC50 > 100000 nM T94324 CO57GS 44138033 IC50 = 5430 nM T94324 CQ2VD5 44219634 IC50 = 250 nM T94324 CIO34V 44564642 Ki = 23 nM T94324 CMA3R6 44574139 IC50 = 254 nM T94324 C5KLR7 44574177 IC50 > 30000 nM T94324 CFS49I 44574178 IC50 > 30000 nM T94324 CJ32DK 44574179 IC50 > 30000 nM T94324 CQOS28 44574180 IC50 = 471 nM T94324 C3RY9V 44574208 IC50 = 13300 nM T94324 CA6Q9Y 44592060 IC50 = 6100 nM T94324 C5H8RA 44598536 IC50 = 150 nM T94324 C42SJP 45141750 IC50 = 503 nM T94324 CLE9U5 45141751 IC50 = 649 nM T94324 CSM1O6 45271073 IC50 = 73000 nM T94324 C2M4GV 46179732 IC50 = 9.8 nM T94324 CS75CD 46179779 IC50 = 6.8 nM T94324 C39YKM 46179780 IC50 = 16.6 nM T94324 C0CKE5 46180624 IC50 > 30000 nM T94324 C7GYH0 46180758 IC50 = 32.8 nM T94324 C27IKH 46180759 IC50 = 10.7 nM T94324 CSC1Y9 46180760 IC50 = 14.5 nM T94324 C70FSJ 46180763 IC50 = 5.8 nM T94324 CQ69AM 46205433 IC50 = 374 nM T94324 CQTI31 46881225 IC50 > 30000 nM T94324 CPSI47 46890583 Ki = 9 nM T94324 C90NYX 46896338 IC50 = 3400 nM T94324 C43TPV 46918824 IC50 = 1995.26 nM T94324 CXH64A 46918825 IC50 = 199.53 nM T94324 C6GY9I 46934544 IC50 = 9050 nM T94324 C3OD2Y 46934546 IC50 = 23900 nM T94324 CL7PS1 49831258 IC50 > 50000 nM T94324 CI5L2P 49846123 IC50 = 1462.81 nM T94324 C4DL0M 49847150 IC50 = 51.6 nM T94324 CC7Y9U 49850262 IC50 = 12.59 nM T94324 C50PXU 49855444 IC50 > 50000 nM T94324 CL7X3K 50898671 IC50 = 501.19 nM T94324 C7MO2J 53325871 IC50 = 3.7 nM T94324 C78GKN 53361474 IC50 = 140 nM T94324 CNB63X 53361475 IC50 = 776 nM T94324 CQ43VH 53363518 Ki = 18 nM T94324 C6Y2EV 53374826 IC50 = 6320 nM T94324 C5A7MU 54613496 IC50 = 3 nM T94324 C7R9TZ 56663191 IC50 = 0.5 nM T94324 CZ25SN 56935695 IC50 > 30000 nM T94324 CA5Q6O 58147189 IC50 > 50000 nM T94324 C4DYC0 58147224 IC50 > 50000 nM T94324 CMP04X 58147302 IC50 > 50000 nM T94324 CLD40J 58465708 IC50 = 41000 nM T94324 C1MB4Q 59323957 IC50 > 30000 nM T94324 CK6LX0 59454220 IC50 = 5000 nM T94324 C2SDN1 59454252 IC50 = 1600 nM T94324 CB7X2E 60151224 IC50 = 37.4 nM T94324 CY05OU 60151225 IC50 = 751 nM T94324 CWO8H0 60152596 IC50 = 1930 nM T94324 CXW14A 60164619 IC50 = 630.96 nM T94324 C7FI3C 60164834 IC50 = 19.95 nM T94324 C9A0HY 60164937 IC50 = 63.1 nM T94324 CBN3L0 69950064 Ki > 10000 nM T94324 C6RFQ8 70676597 IC50 > 20000 nM T94324 CQY1I6 70789579 Ki > 10000 nM T94324 C6KBD4 71534512 IC50 = 14 nM T94324 CT51EW 71534810 IC50 = 4 nM T94324 C7QN3O 71534812 IC50 = 1 nM T94324 C8M3HU 71537640 IC50 = 7 nM T94324 C2QML7 71537641 IC50 = 5 nM T94324 CZJX53 71537927 IC50 = 6000 nM T94324 CU0ZE6 71537928 IC50 = 11 nM T94324 CH9FS7 71537929 IC50 = 81 nM T94324 CTW95A 71537931 IC50 = 11 nM T94324 C3C0RO 71538475 IC50 = 6 nM T94324 CIA28E 71538746 IC50 = 11 nM T94324 CFCV26 71538748 IC50 = 658 nM T94324 CY2T1Q 71538749 IC50 = 310 nM T94324 C4A6VJ 71538750 IC50 = 9 nM T94324 CG72NC 71538751 IC50 = 14 nM T94324 C7MW4N 71582992 IC50 = 316.23 nM T94324 CKR6U8 71583101 IC50 = 21000 nM T94324 CBZ5S9 71583103 IC50 = 7700 nM T94324 C3PSJ9 71583105 IC50 = 5900 nM T94324 CU3N9R 71811227 IC50 = 17500 nM T94324 C0MV3O 71811291 IC50 > 10000 nM T94324 C7UYD4 71811292 IC50 = 5140 nM T94324 C7XL3N 71811293 IC50 = 29800 nM T94324 CI9H6L 72164895 IC50 = 51 nM T94324 CS5UL7 72195322 IC50 = 94 nM T94324 CV09DJ 72734543 IC50 = 5000 nM T94324 CS6LW0 72946640 IC50 = 51 nM T94324 CXM37Z 72946641 IC50 = 93 nM T94324 CQA16N 72946833 IC50 = 113 nM T94324 CNR7Z2 72946834 IC50 = 244 nM T94324 C12JYS 72946835 IC50 = 147 nM T94324 C5Y9XH 72946836 IC50 = 88 nM T94324 CVZR94 72946837 IC50 = 6830 nM T94324 C8-AUG 72946838 IC50 = 227 nM T94324 CHQ39Y 72947043 IC50 = 125 nM T94324 CCST90 72947044 IC50 = 30 nM T94324 C7J3RH 72947045 IC50 = 163 nM T94324 CX3W1T 73333311 IC50 = 3700 nM T94324 C68LBO 73349131 IC50 = 6 nM T94324 CXK86S 73355189 IC50 = 70 nM T94324 C3UC9H 73891099 IC50 = 8400 nM T94324 CL4JQ3 76331862 IC50 = 4890 nM T94324 C08CPW 76335428 IC50 = 210 nM T94324 C06YBD 86302594 IC50 = 886 nM T94324 C6M9PL 86765212 IC50 = 4130 nM T94324 CS5I4Y 87261507 IC50 = 290 nM T94324 C2U9LW 88981186 IC50 = 1000 nM T94324 CB47VC 89464167 IC50 = 2930 nM T94324 CYW51P 90654946 IC50 = 63900 nM T94324 CJH1S6 90654947 IC50 > 100000 nM T94324 CSR56C 90655296 IC50 = 3220 nM T94324 CSDO81 90664458 Ki = 23 nM T94324 CJO6T1 91810840 IC50 = 700 nM T94324 CYJ12Q 91884636 IC50 = 11 nM T94324 C34WIG 92045024 IC50 > 100000 nM T94324 C9OC0F 101882265 IC50 = 71100 nM T94324 C2I8XR 101882814 Ki = 4000 nM T94324 C8KZB4 101883993 Ki = 700 nM T94324 C7Q6ID 101884982 IC50 = 15 nM T94324 CR46PQ 101884983 IC50 = 32 nM T94324 CRZ83C 101884989 IC50 = 40 nM T94324 CT7Z8F 102514716 IC50 = 78310 nM T94324 CSU52M 118656852 IC50 = 6400 nM T94324 CB6AJ9 118656853 IC50 = 13000 nM T94324 C45UYG 118709095 IC50 = 85000 nM T94324 C7QHE4 118712502 IC50 = 0.2 nM T94324 C8KSD6 118712503 IC50 = 0.5 nM T94324 C1JFZ7 118714371 IC50 = 774 nM T94324 CXF0U3 118714375 IC50 = 136 nM T94324 C2M5OR 118714376 IC50 = 25 nM T94324 CY4GN9 118714377 IC50 = 29 nM T94324 CM5QT7 118719376 Ki = 1600 nM T94324 CPB7C3 118719377 Ki = 700 nM T94324 C09OGH 118719378 Ki = 600 nM T94324 CR5VC1 118719379 Ki = 1000 nM T94324 C32LCM 118719380 Ki = 300 nM T94324 C8U6YR 118719381 Ki = 170 nM T94324 C9Y0HV 118719382 Ki = 300 nM T94324 CY0J4D 118719383 Ki = 230 nM T94324 CCYU59 118719817 IC50 = 7 nM T94324 CMV2W9 118721625 IC50 = 9 nM T94324 CF5TO3 118721859 IC50 = 116 nM T94324 CK97TZ 118721860 IC50 = 5 nM T94324 CYV30O 118721861 IC50 = 4 nM T94324 C5WYI1 118721862 IC50 = 2 nM T94324 CSMW25 118721863 IC50 = 1170 nM T94324 C5B1KM 118721864 IC50 = 189 nM T94324 CG8LZ0 118721865 IC50 = 6290 nM T94324 CPCN23 118721866 IC50 = 2990 nM T94324 CM0A9U 118721867 IC50 = 3930 nM T94324 CI8G4X 118737400 IC50 = 1800 nM T94324 C5L8QM 118884518 IC50 = 39500 nM T94324 CIA40K 121472983 IC50 = 33000 nM T94324 C28JVO 122192004 IC50 = 138 nM T94324 CF2D8U 122192005 IC50 = 395 nM T94324 C3V5ND 122550211 IC50 = 1176 nM T94324 CZE35C 122648343 IC50 = 6.85 nM T94324 C54RNT 122648367 IC50 = 2.8 nM T94324 C1UVI7 122648600 IC50 = 17.55 nM T94324 CMX59K 122648648 IC50 = 2.83 nM T94324 CVZ64I 122648649 IC50 = 0.86 nM T94324 CV9I8D 127030313 IC50 = 10200 nM T94324 C8IEV4 130258911 IC50 = 1510 nM T94324 C6OXE3 132134663 IC50 = 80 nM T94324 C6X3HG 132145728 IC50 = 1256 nM T94324 C8O9DP 132157820 IC50 = 9791 nM T94324 C4KE3N 132938351 IC50 > 10000 nM T94324 C05FVT 134492522 IC50 > 10000 nM T94324 CT19ND 136110961 IC50 > 100000 nM T94324 CY9U0E 136173089 IC50 = 40 nM T94324 C67EFJ 137628684 IC50 = 0.58 nM T94324 C1V8QE 137634156 IC50 = 5.012 nM T94324 C6JVG9 137635398 IC50 = 19 nM T94324 CGK2M9 137649620 IC50 = 3.6 nM T94324 C5FHD3 137652442 IC50 = 20400 nM T94324 CCR5B3 137654793 IC50 = 31 nM T94324 C1SBN5 137654946 IC50 = 8230 nM T94324 C76OGQ 137656942 IC50 = 10000 nM T94324 CEJI95 137661885 IC50 = 21 nM T94324 CAQ62X 137701235 Ki = 3 nM T94324 C7EM3I 138393071 IC50 = 59800 nM T94324 CN2UH1 139303146 IC50 = 1.98 nM T94324 C7XI0V 141764754 IC50 = 102 nM T94324 CX0E9B 142505968 IC50 = 16900 nM T94324 CBJC50 142505992 IC50 = 33730 nM T94324 CKBF56 142506033 IC50 = 2073 nM T94324 CGNQ74 142506189 IC50 = 14700 nM T94324 C1T3IQ 142506210 IC50 = 1502 nM T94324 CKG98W 145953085 IC50 = 1870 nM T94324 CK1XI0 145960971 IC50 > 10000 nM T94324 C3PWD4 145964064 IC50 = 7050 nM T94324 CEDK05 145964533 IC50 = 15500 nM T94324 CDY56B 145964885 IC50 = 5890 nM T94324 CJAE67 145966594 IC50 > 100000 nM T94324 C19POY 145967140 IC50 = 47900 nM T94324 CSJ81Y 145968726 IC50 = 5240 nM T94324 CI43DY 145970786 IC50 > 100000 nM T94324 C4HTO2 145973543 IC50 = 8240 nM T94324 CVM0Z3 145974125 IC50 > 100000 nM T94324 C8YEJ9 145974425 IC50 > 100000 nM T94324 CE8I5V 145975869 IC50 = 7740 nM T94324 CMUA94 145976675 IC50 = 9100 nM T94324 CN6UO4 145977003 IC50 > 100000 nM T94324 CKAQ67 145977127 IC50 = 18900 nM T94324 COR40V 145978805 IC50 > 100000 nM T94324 CIM41N 145980574 IC50 = 9.12 nM T94324 CMB08D 145981960 IC50 = 2910 nM T94324 CWD0A9 145983712 Ki = 1.2 nM T94324 C56MWZ 145986208 Ki = 50 nM T94324 CS79CE 145986632 IC50 = 7.55 nM T94324 C82CIN 145988785 IC50 > 30000 nM T94324 C0GMR1 146585718 IC50 = 9996 nM T94324 CB7K1M 146676960 IC50 = 79.43 nM T94324 C0YXS8 147254231 IC50 = 4997 nM T94324 CN71OS 149405396 IC50 = 1470 nM T94324 C9FIY4 153534005 IC50 = 923 nM T94324 CA1J3N 155517086 IC50 = 268 nM T94324 CY54TU 155518062 IC50 = 13000 nM T94324 CEH2N5 155518106 IC50 = 164 nM T94324 CMDR68 155518334 IC50 = 125.89 nM T94324 CDY5H6 155519645 IC50 > 10000 nM T94324 CAZ3S7 155521187 IC50 = 9400 nM T94324 CZ75FW 155521272 IC50 = 114 nM T94324 C63NOC 155527045 IC50 = 10000 nM T94324 CZMC49 155530597 IC50 = 2.1 nM T94324 C8IMN6 155533398 IC50 = 5011.87 nM T94324 CIZ46A 155533876 IC50 = 14000 nM T94324 CPE68B 155534222 IC50 = 15.85 nM T94324 C6LB5D 155535084 IC50 > 30000 nM T94324 CTF98X 155537473 IC50 = 320 nM T94324 CLD19W 155539311 IC50 = 2670 nM T94324 CK45LA 155546486 IC50 = 630.96 nM T94324 C3HB0U 155546555 IC50 = 5.012 nM T94324 CS3GO2 155546558 IC50 = 660 nM T94324 C93ZWM 155546700 IC50 = 158.49 nM T94324 CE0YL6 155549538 IC50 = 3000 nM T94324 CA03BO 155551057 IC50 = 25.12 nM T94324 CV4Y5B 155552792 IC50 = 5300 nM T94324 CGDF76 155554360 IC50 = 10000 nM T94324 CC56ED 155554844 IC50 = 5.7 nM T94324 CXGR50 155555191 IC50 > 30000 nM T94324 CFW90N 155555562 IC50 = 1.43 nM T94324 CIN57Q 155556138 IC50 = 2690 nM T94324 C8AUB0 155558567 IC50 = 950 nM T94324 CPD50Q 155559583 IC50 = 1600 nM T94324 C87JXN 155564870 IC50 = 3.981 nM T94324 CZDC03 155565491 IC50 > 30000 nM T94324 CW5XB4 155569484 IC50 = 2910 nM T94324 D00GBB 11449246 Ki = 40 nM T94324 D00SEE 11379392 IC50 = 270 nM T94324 D01YBR 44591988 IC50 = 7840 nM T94324 D04KQF 6675804 Ki = 373.7 nM T94324 D05OVV 11993691 IC50 = 870 nM T94324 D09RKA 72946782 IC50 = 5000 nM T94324 D0B3ZM 11436024 IC50 = 1220 nM T94324 D0E9DD 16095101 Ki = 20 nM T94324 D0K7QR 45269423 IC50 = 250 nM T94324 D0N9AK 44138031 IC50 = 7360 nM T94324 D0Q5DI 71462653 IC50 = 100 nM T94324 D0Q5MC 24753719 IC50 = 13000 nM T94324 D0Q9PO 16095114 Ki = 10 nM T94324 D0T0SK 44138032 IC50 = 1580 nM T94324 D0XZ9Q 11149404 IC50 = 252 nM T94324 D0Z8PX 24757913 IC50 = 2210 nM T98062 D0B3HD 2519 IC50 = 114000 nM T98062 D0LF1U 5287969 IC50 = 1000 nM T98062 C8IJ0B 79025 Ki = 1700000 nM T98062 C8WA2E 3658622 IC50 ~ 100000 nM T98062 C8BDA7 4369162 Ki = 5100 nM T98062 C0E9MB 9840862 IC50 = 14 nM T98062 CWS9P8 9931451 IC50 = 6000 nM T98062 CDZ2L0 9953189 IC50 = 50000 nM T98062 COL4X7 9954417 IC50 = 60 nM T98062 C65DJK 9958633 IC50 = 11 nM T98062 C5BAT1 10043666 IC50 = 55 nM T98062 CC4IR6 10125909 IC50 = 38 nM T98062 CA3TJ8 10409816 IC50 = 50000 nM T98062 CZR8W9 10477826 IC50 = 138 nM T98062 C8V9TB 11187969 IC50 = 120 nM T98062 CMI72Q 11200159 IC50 = 190 nM T98062 CL4JZ8 11200978 IC50 > 200000 nM T98062 CXRG64 11222164 IC50 = 110 nM T98062 C3C2JH 11292222 IC50 = 110 nM T98062 C1VH7I 11324538 IC50 = 2500 nM T98062 C1W7PG 11337343 IC50 = 200 nM T98062 CKZ57R 11338774 IC50 = 140 nM T98062 CW3C9Z 11451272 IC50 = 710 nM T98062 CXH6R7 11465977 IC50 = 350 nM T98062 CY0IT9 11475200 IC50 = 280 nM T98062 CKO62P 11475654 IC50 = 320 nM T98062 CP0XI8 11772828 IC50 = 730 nM T98062 CP56TC 11774080 IC50 = 190 nM T98062 CUC7N2 11785069 IC50 = 420 nM T98062 CY1J3I 13908996 Ki = 1000000 nM T98062 CI0JH1 19002057 Ki = 1.6 nM T98062 CDM7V9 21974595 IC50 = 32 nM T98062 CIK5V6 44342320 IC50 = 41 nM T98062 COZG47 44342348 IC50 = 12.9 nM T98062 C49TDU 44342362 IC50 = 52 nM T98062 CF8D0Y 44342363 IC50 = 15000 nM T98062 C30MEI 44342377 IC50 = 1195 nM T98062 CASE46 44342459 IC50 = 178 nM T98062 C25DBF 44342460 IC50 = 8.28 nM T98062 CQH1X0 44342462 IC50 = 10.61 nM T98062 CX2G3N 44342474 IC50 = 29 nM T98062 CNX08S 44342475 IC50 = 10 nM T98062 CXEC30 44342489 IC50 = 37 nM T98062 CK84CQ 44342512 IC50 = 91 nM T98062 C6M3LQ 44342540 IC50 = 185 nM T98062 C5R3WV 44342585 IC50 = 233 nM T98062 CA3G4I 44342602 IC50 = 6 nM T98062 CX15TC 44342751 IC50 = 26 nM T98062 CLZD72 44342773 IC50 = 19.9 nM T98062 CT1GA3 44345051 Ki = 11 nM T98062 CDS4A6 44345146 Ki = 3000 nM T98062 CY8L5Q 44354084 IC50 = 647 nM T98062 CVY98H 44354099 IC50 = 109 nM T98062 C0C2IS 44354283 IC50 = 12300 nM T98062 CX7TL1 44354301 IC50 = 29 nM T98062 CE65JT 44354322 IC50 = 167 nM T98062 CINT36 44354348 IC50 = 468 nM T98062 C8UCM7 44354349 IC50 = 200 nM T98062 CNR06G 44354350 IC50 = 181 nM T98062 CT43DB 44354362 IC50 = 844 nM T98062 C1EIY4 44354370 IC50 = 110 nM T98062 CHGM26 44354391 IC50 = 9 nM T98062 CI03FC 44354408 IC50 = 1860 nM T98062 CRXN57 44354446 IC50 = 25 nM T98062 CDE41K 44354454 IC50 = 80 nM T98062 CQ9IP7 44354455 IC50 = 57 nM T98062 CHTI61 44354456 IC50 = 140 nM T98062 CS7CE9 44354829 IC50 = 12 nM T98062 CIQM91 44354843 IC50 = 3 nM T98062 CU60QX 44354844 IC50 = 12 nM T98062 C4OX0H 44357872 IC50 = 98 nM T98062 CE36PI 44357873 IC50 = 89 nM T98062 C6UIG5 44357874 IC50 = 73 nM T98062 C7B6LO 44357907 IC50 = 56 nM T98062 CSEP-56 44357919 IC50 = 105 nM T98062 CS2VR8 44357925 IC50 = 83 nM T98062 CV4CE2 44357926 IC50 = 39 nM T98062 CZ3LM4 44357933 IC50 = 240 nM T98062 CTCI46 44357937 IC50 = 57 nM T98062 CS20RO 44357938 IC50 = 58 nM T98062 C3ZR9I 44358037 IC50 > 20000 nM T98062 C85KUT 44358038 IC50 = 550 nM T98062 CGEX65 44358070 IC50 = 2700 nM T98062 C6WE2Q 44358094 IC50 = 110 nM T98062 C8JV9Q 44358107 IC50 = 1700 nM T98062 CE3PV5 44358108 IC50 = 850 nM T98062 C6KXF8 44358150 IC50 = 2100 nM T98062 CBJ6P0 44358151 IC50 = 88 nM T98062 C20AUQ 44358152 IC50 > 20000 nM T98062 C3YGV2 44358155 IC50 = 69 nM T98062 C8EFT0 44358159 IC50 = 2440 nM T98062 CQ4RA3 44358172 IC50 > 20000 nM T98062 CGK1A5 44358173 IC50 = 6800 nM T98062 CTPE57 44358204 IC50 = 55 nM T98062 C3EW8Q 44358205 IC50 > 20000 nM T98062 CAK56U 44358343 IC50 = 2310 nM T98062 C65TFS 44358344 IC50 = 21700 nM T98062 CU7OF1 44358402 IC50 = 120 nM T98062 CT6J1N 44403045 IC50 = 2500 nM T98062 C9B7FV 44403049 IC50 = 5000 nM T98062 CT7JL5 44403050 IC50 > 10000 nM T98062 CT31XP 44403051 IC50 = 2500 nM T98062 CL6T2G 44403054 IC50 > 10000 nM T98062 C01GJK 44403058 IC50 = 480 nM T98062 C51UIK 44403142 IC50 > 10000 nM T98062 C6V2QU 44403153 IC50 = 160 nM T98062 CY03FE 44403159 IC50 > 10000 nM T98062 C12BMA 44403167 IC50 = 5700 nM T98062 C1Q0HV 44403170 IC50 = 710 nM T98062 C2FBL6 44403171 IC50 = 580 nM T98062 CG06DV 46905967 IC50 > 10000 nM T98062 CE94YF 52946782 Ki = 4600 nM T98062 CE41UW 56603813 Ki = 1020 nM T98062 C01YUK 56603814 Ki = 3270 nM T98062 C8N0LT 56603815 Ki = 1940 nM T98062 CD0U1K 57519731 IC50 = 291400 nM T98062 CS8NM0 118719323 Ki = 4200 nM T98062 D01BZE 73659 IC50 = 28000 nM T98062 D0E4SM 657140 IC50 = 900 nM T98062 D0F9RO 6918774 IC50 = 20000 nM T98062 D0S0AN 444746 IC50 = 500 nM T36806 C4FQ8G 10214423 IC50 = 1920 nM T36806 CK7F4Q 46849717 IC50 = 4280 nM T36806 C92VFP 46849884 IC50 = 4500 nM T36806 C38SPE 46850575 IC50 = 17000 nM T36806 C1OJ9B 54588038 IC50 = 5980 nM T36806 C04LVP 54588438 IC50 = 240 nM T36806 CPU82S 54588586 IC50 = 1710 nM T36806 C8F6ZL 54588588 IC50 = 420 nM T36806 CU0JG3 54588590 IC50 = 600 nM T36806 C7B5AK 54588591 IC50 = 2560 nM T36806 CX6HJ9 54588725 IC50 = 270 nM T36806 CAF89Z 66832756 IC50 = 290 nM T36806 C03CMO 66832782 IC50 = 1100 nM T36806 C6SFG4 66832803 IC50 = 3720 nM T36806 C7UPK5 66832944 IC50 = 340 nM T36806 CW0Q7C 66832969 IC50 = 70 nM T36806 CN1WR8 66833017 IC50 = 50 nM T36806 CLE15I 66833072 IC50 = 980 nM T36806 CED5U9 66833182 IC50 = 640 nM T36806 CLVS71 66833213 IC50 = 509 nM T36806 CK3CI7 66833351 IC50 = 230 nM T36806 CI87XR 66833376 IC50 = 620 nM T36806 CI7B1J 66833380 IC50 = 230 nM T36806 C1LD9T 66833489 IC50 = 4020 nM T36806 CR3D1L 66833558 IC50 = 330 nM T36806 C3JT0R 68064421 IC50 > 300000 nM T36806 C0XL8K 71554360 IC50 = 30 nM T36806 CY9U5M 71554361 IC50 = 23 nM T36806 CZ6DY1 71554539 IC50 = 85 nM T36806 C6X4NP 71554627 IC50 = 47 nM T36806 C93EFD 71554628 IC50 = 33 nM T36806 C7U0GH 71554631 IC50 = 390 nM T36806 COR30T 71554632 IC50 = 320 nM T36806 CAB0X2 71554633 IC50 = 190 nM T36806 C9O1DZ 71579993 IC50 = 4600 nM T36806 C7TOP2 71579996 IC50 = 57000 nM T36806 C2IDG5 71579997 IC50 = 6440 nM T36806 CUY30S 71600432 IC50 = 67 nM T36806 CYP9J5 71600433 IC50 = 1090 nM T36806 C4VZ5F 71600434 IC50 = 310 nM T36806 CC7O3P 71600564 IC50 = 550 nM T36806 CG4I0J 71678226 IC50 = 934 nM T36806 CM05JI 71716534 IC50 = 1350 nM T36806 C4O6DF 71719961 IC50 = 1920 nM T36806 C4KC0N 71720821 IC50 = 15500 nM T36806 CVHJ68 71818258 IC50 = 4650 nM T36806 CZ8S5P 71818259 IC50 = 1120 nM T36806 CZIO09 145983883 Ki = 322000 nM T36806 C7N6LU 145983954 Ki = 437000 nM T36806 CN6QR9 46849719 IC50 = 5070 nM T36806 D08PUJ 9793992 Ki = 8.5 nM T36806 D0YY4Y 446124 Ki = 51 nM T34239 C60HDK 29732 Ki = 2930 nM T34239 CO85ZP 44073 Ki = 1710 nM T34239 CX20NK 86369 Ki = 720 nM T34239 CB45IQ 231239 Ki = 87096.36 nM T34239 CTRY20 45276320 Ki = 10232.93 nM T34239 C12OZY 45276488 Ki = 330 nM T34239 CDC29W 45276489 Ki = 250 nM T34239 CBKQ57 45276490 Ki = 1000 nM T34239 CH80QR 45276491 Ki = 831.76 nM T34239 CO6B9G 45276492 Ki = 1070 nM T34239 CE9JR2 45276493 Ki = 2020 nM T34239 CGE71M 45276494 Ki = 1690 nM T34239 CDR23M 45276651 Ki = 3090.3 nM T34239 CSB27P 45276652 Ki = 1348.96 nM T34239 CKN23D 45276653 Ki = 2170 nM T34239 CUV32Q 45276654 Ki = 977.24 nM T34239 CU97ZM 45276655 Ki = 8610 nM T34239 CFV0T7 45276656 Ki = 3981.07 nM T34239 CL9D6W 45276657 Ki = 720 nM T34239 C6KAJ2 45276811 Ki = 720 nM T34239 C4EZ9R 45276812 Ki = 1580 nM T34239 CJ59ZF 45276813 Ki = 1584.89 nM T34239 C2BR9F 45276814 Ki = 15848.93 nM T34239 CX57BU 45276815 Ki = 320 nM T34239 CL3W4D 45276816 Ki = 360 nM T34239 CJX87S 45276817 Ki = 1540 nM T34239 C85MWX 45276964 Ki = 700 nM T34239 COB49Y 45276965 Ki = 10920 nM T34239 C0NSA5 45276966 Ki = 1412.54 nM T34239 C0NOL8 45276967 Ki = 7413.1 nM T34239 CT2W4V 45276968 Ki = 1170 nM T34239 C60NMO 45276969 Ki = 6918.31 nM T34239 C5NB3K 45276970 Ki = 7413.1 nM T34239 CJM64K 45277123 Ki = 5970 nM T34239 C0GHU9 45277124 Ki = 5830 nM T34239 C5ZBW4 45277125 Ki = 8128.31 nM T34239 CKRV71 45277126 Ki = 1690 nM T34239 CATO69 45277127 Ki = 3090.3 nM T34239 CC4U8W 45277128 Ki = 11120 nM T34239 C8P4XM 45277129 Ki = 18620.87 nM T34239 C4JVH2 56837415 Ki = 40 nM T34239 CR70BZ 57390531 Ki = 1260 nM T34239 CE64BC 57390532 Ki = 9730 nM T34239 C4HUZ9 57390533 Ki = 5820 nM T34239 CG1YD2 57392291 Ki = 17700 nM T34239 CN5ZC6 57392297 Ki = 340 nM T34239 CF8PJ0 57392298 Ki = 5890 nM T34239 C9EBG8 57392299 Ki = 8670 nM T34239 COEV07 57392300 Ki = 34400 nM T34239 CH40BM 57392301 Ki = 43500 nM T34239 C91YDX 57394052 Ki = 9260 nM T34239 CW1J8N 57394053 Ki = 1280 nM T34239 C5UT1F 57394054 Ki = 21400 nM T34239 CZJU03 57394055 Ki = 173000 nM T34239 C2XYE9 57394116 Ki = 1920 nM T34239 C27FLP 57395813 Ki = 200 nM T34239 CB13FP 57395814 Ki = 12000 nM T34239 C7UXS9 57397594 Ki = 27500 nM T34239 CN84DI 57397602 Ki = 1580 nM T34239 CO5NK6 57399270 Ki = 3050 nM T34239 CCJ30H 57399271 Ki = 1310 nM T34239 CEO83Q 57399272 Ki = 20700 nM T34239 C0JSC5 57401037 Ki = 3460 nM T34239 CPE49M 57401038 Ki = 15600 nM T34239 CVQZ75 57401039 Ki = 245000 nM T34239 C6ORQ1 76308283 Ki = 19350 nM T34239 CSW09X 76311931 Ki = 15135.61 nM T34239 CN7CL1 76315474 Ki = 776.25 nM T34239 CZ7GD2 76315475 Ki = 8128.31 nM T34239 CJ76IW 76315476 Ki = 47863.01 nM T34239 CCEM92 76315477 Ki = 63095.73 nM T34239 C5H2UA 76315478 Ki = 27542.29 nM T34239 CXY12J 76319155 Ki = 120 nM T34239 C2O0JW 76319156 Ki = 41350 nM T34239 C5SE2N 76319157 Ki = 1023.29 nM T34239 CE10ZQ 76319158 Ki = 130970 nM T34239 C8JD7L 76322810 Ki = 300 nM T34239 C38TNH 76322811 Ki = 95 nM T34239 CS49CH 76322812 Ki = 7413.1 nM T34239 CE8K5O 76322813 Ki = 354813.39 nM T34239 C46XKD 76322814 Ki = 4466.84 nM T34239 CWN0A4 76326377 Ki = 1023.29 nM T34239 C5AJV8 76329991 Ki = 670 nM T34239 C12OQD 76329992 Ki = 524.81 nM T34239 C2Y4WQ 76333625 Ki = 199.53 nM T34239 CAZ2H8 76333626 Ki = 66069.34 nM T34239 C8OS2E 76333627 Ki = 33113.11 nM T34239 COGF10 76333628 Ki = 7020 nM T34239 C7THY0 76333629 Ki = 3300 nM T34239 CU7OI5 76333630 Ki = 24547.09 nM T34239 CXF57Q 76333631 Ki = 47350 nM T34239 CN7WI8 76333632 Ki = 123026.88 nM T34239 CKL0Y7 76333633 Ki = 44830 nM T34239 CZX45A 76333634 Ki = 690 nM T37384 D0WS1V 448991 IC50 = 1200 nM T37384 CGAN35 2856 IC50 = 7000 nM T37384 CKIW13 10428636 IC50 > 500000 nM T37384 CM9ZG4 135965879 IC50 > 33000 nM T37384 D02XHC 448912 IC50 = 2500 nM T37384 D03EIM 6436801 IC50 = 24000 nM T37384 D07OAT 456214 IC50 = 80 nM T79326 CN74UD 611792 IC50 = 319000 nM T79326 C7VN1X 698057 IC50 = 319000 nM T79326 C02EUQ 49800098 IC50 < 5000 nM T79326 CP0U6G 53348215 IC50 = 2400 nM T79326 C0SWH5 53348216 IC50 = 12 nM T79326 CNKU96 53348217 IC50 = 270 nM T79326 C6CVN9 53379388 IC50 = 590 nM T79326 CI0V4P 53379389 IC50 = 920 nM T79326 CMR98W 53494134 IC50 = 670 nM T79326 CM62SE 53494135 IC50 = 34 nM T79326 C9P7VJ 53494875 IC50 = 7 nM T79326 CV13ZT 53494876 IC50 = 8 nM T79326 C2K7XI 53494877 IC50 = 7.1 nM T79326 CIUE20 56659792 IC50 = 80 nM T79326 C70CKM 56659840 IC50 = 830 nM T79326 C8ZN6L 56659841 IC50 = 23 nM T79326 C1ZFD0 56659842 IC50 = 160 nM T79326 CBQP98 56663308 IC50 = 220 nM T79326 CTF31E 56663309 IC50 = 11500 nM T79326 C35ZNW 56663310 IC50 = 1680 nM T79326 C3Z0AY 56663311 IC50 = 4520 nM T79326 CP72DX 56663312 IC50 = 940 nM T79326 C0OZQ7 56666738 IC50 = 42 nM T79326 CV9ZF3 56666739 IC50 = 9800 nM T79326 C2T0AQ 56666741 IC50 > 20000 nM T79326 CKZ3F4 56670113 IC50 = 710 nM T79326 C0TGL2 56670164 IC50 = 40 nM T79326 CN18PK 56670165 IC50 = 570 nM T79326 CVF27X 56670166 IC50 = 680 nM T79326 C9GO2M 56673627 IC50 = 710 nM T79326 CP7YS5 56673684 IC50 = 680 nM T79326 CGS4B0 56673685 IC50 = 240 nM T79326 CM84TQ 56673686 IC50 = 11500 nM T79326 C8QHX4 56673687 IC50 = 3520 nM T79326 C6CH5P 56676999 IC50 = 590 nM T79326 CDJ0S5 56677000 IC50 = 87 nM T79326 CQH7W1 56677001 IC50 = 1280 nM T79326 C6TIA9 56677002 IC50 = 1380 nM T79326 C84KRQ 56680270 IC50 = 330 nM T79326 CPS5Y1 56680271 IC50 = 560 nM T79326 CQU60O 56680272 IC50 > 10000 nM T79326 CD1CI4 56680273 IC50 = 440 nM T79326 CRS85L 56680332 IC50 = 480 nM T79326 CIM4E7 56680333 IC50 = 3200 nM T79326 C5S6AJ 56683597 IC50 = 310 nM T79326 CQHN29 56683647 IC50 = 380 nM T79326 CNC9I5 56683648 IC50 = 560 nM T79326 CUT2V8 56683649 IC50 = 860 nM T79326 CTV34J 56683650 IC50 = 1280 nM T79326 C0DC9Z 66552359 IC50 = 70 nM T79326 CFDO28 66552360 IC50 = 58 nM T79326 CC75UP 66552361 IC50 = 110 nM T79326 CIX3Z7 66552362 IC50 = 40 nM T79326 CBJR84 66552363 IC50 = 66 nM T79326 C23MYW 66552422 IC50 = 4600 nM T79326 CI6C3N 66552424 IC50 = 6000 nM T79326 CM32WU 66552425 IC50 = 43 nM T79326 CK6LN3 66552476 IC50 = 2 nM T79326 CDW6R9 66552477 IC50 = 15 nM T79326 CK6WO0 66552478 IC50 = 48 nM T79326 C7H8BO 66552479 IC50 = 28 nM T79326 C17MVF 66552480 IC50 = 50 nM T79326 C2ADI8 66552529 IC50 = 30 nM T79326 CM4X2Z 70681158 IC50 = 400 nM T79326 CW46XO 70681159 IC50 = 2800 nM T79326 CT0EJ4 70681160 IC50 = 100 nM T79326 C63DRQ 70681161 IC50 = 1500 nM T79326 C9N3IU 70681162 IC50 = 540 nM T79326 C1YK6X 70681163 IC50 > 9000 nM T79326 C7HM6T 70681164 IC50 = 2300 nM T79326 CZG8H1 70681165 IC50 = 400 nM T79326 CC61JR 70681166 IC50 = 60 nM T79326 CFH0B9 70683270 IC50 > 9000 nM T79326 C04TSR 70684418 IC50 = 800 nM T79326 CNO8A6 70685368 IC50 = 3200 nM T79326 CD0R6N 70685369 IC50 = 2000 nM T79326 CREQ90 70685370 IC50 = 3000 nM T79326 CH16UP 70685371 IC50 = 5000 nM T79326 C5QU9J 70685372 IC50 = 380 nM T79326 C2SCV9 70685373 IC50 > 9000 nM T79326 CV5OT0 70685374 IC50 = 23 nM T79326 C69NGQ 70685375 IC50 = 140 nM T79326 C76GVU 70685376 IC50 = 110 nM T79326 CT7Y5I 70687508 IC50 > 9000 nM T79326 C5YFU7 70687509 IC50 = 200 nM T79326 CS1P0O 70688677 IC50 = 440 nM T79326 CQ3GO2 70689564 IC50 = 130 nM T79326 CT4J8P 70689565 IC50 = 70 nM T79326 C7ZPE6 70689566 IC50 = 18 nM T79326 CXWJ01 70689567 IC50 = 18 nM T79326 C2F4IH 70689568 IC50 = 10 nM T79326 C6HTO7 70691688 IC50 = 400 nM T79326 CM2K4B 70691689 IC50 = 1700 nM T79326 C07WDJ 70691690 IC50 = 300 nM T79326 C19LIP 70691691 IC50 = 300 nM T79326 CP2A0Y 70691692 IC50 > 7000 nM T79326 CH95TU 70691693 IC50 = 710 nM T79326 C0ABZ9 70691694 IC50 = 50 nM T79326 CE1IG0 70691695 IC50 = 30 nM T79326 C75YBN 70691696 IC50 = 130 nM T79326 CW6XI0 70693774 IC50 = 200 nM T79326 C83LJW 70693775 IC50 = 170 nM T79326 C29QNW 70693776 IC50 = 1600 nM T79326 C2OV0D 70693777 IC50 = 300 nM T79326 CVMS13 70693778 IC50 = 270 nM T79326 CCF0Y3 70695885 IC50 > 9000 nM T79326 C72JPQ 70695886 IC50 = 1500 nM T79326 C3ZL0K 70695887 IC50 = 30 nM T79326 CB5KD0 70696970 IC50 = 300 nM T79326 C84KFB 88543284 IC50 > 500000 nM T79326 C75NAX 129278694 IC50 = 14 nM T79326 C7N1MJ 129900195 IC50 = 118000 nM T79326 COG0W1 129900198 IC50 = 390 nM T79326 C7GP8M 135985432 IC50 = 6100 nM T79326 CLGQ08 137635756 IC50 = 670 nM T79326 CXJ96U 137639342 IC50 = 1030 nM T79326 CF28YL 137648475 IC50 = 16790 nM T79326 C8G4RL 137654444 IC50 = 23988.33 nM T79326 CPQ26I 137660802 IC50 = 1480 nM T13127 D01GBY 124087 IC50 > 65000 nM T13127 D0X4RS 5745 IC50 = 14000 nM T13127 D07RKN 11539477 IC50 = 53000 nM T13127 D0C2HI 60680 IC50 = 27000 nM T13127 D0Q5VW 216454 IC50 = 2 nM T13127 D0W4HZ 148195 IC50 = 1.9 nM T13127 D0Z1NY 448545 IC50 = 1.3 nM T13127 D03GQH 132887 IC50 = 50000 nM T13127 D04DYZ 447312 EC50 = 16 nM T13127 D0EY9P 9845545 IC50 = 250 nM T13127 D0H5VF 9953221 IC50 = 1.8 nM T13127 D0L5AS 10432334 IC50 = 80 nM T13127 D0N1XD 6223 IC50 = 80000 nM T13127 D0W2ED 54041632 IC50 = 20 nM T13127 C6OZ1C 1267 IC50 = 1.1 nM T13127 C7Y8VS 1318 IC50 = 4000000 nM T13127 CB4Z9P 1474 IC50 = 100000000 nM T13127 CX6EM9 69527 IC50 = 854000 nM T13127 C1F9XW 75110 IC50 > 1000000 nM T13127 CH4QP5 122486 IC50 = 449000 nM T13127 C0IFW4 131994 IC50 = 21000 nM T13127 C8G4BN 300704 IC50 > 100000 nM T13127 C1OCR0 300707 IC50 > 100000 nM T13127 C34GEC 390610 IC50 = 620000 nM T13127 CNJU05 397855 IC50 = 0.9 nM T13127 C9A8BK 447390 IC50 = 0.39 nM T13127 C58YHM 493392 IC50 > 1000000 nM T13127 C18WTL 508167 IC50 = 200 nM T13127 C57QBP 508169 IC50 = 3000 nM T13127 C0MJD5 631421 IC50 = 10950 nM T13127 C4JYU3 644328 IC50 = 6 nM T13127 CBWH59 1097759 IC50 = 6900 nM T13127 CTB2J9 1100763 IC50 = 440 nM T13127 CK3Y8E 1302012 IC50 = 5600 nM T13127 CN7Q5K 1739605 IC50 = 370 nM T13127 CC8FZ5 1807368 IC50 = 2570 nM T13127 CNUY90 1807379 IC50 = 4210 nM T13127 CY3H5W 2814842 IC50 = 5400 nM T13127 CX5J3H 2814844 IC50 = 13350 nM T13127 CHSE90 2819763 IC50 > 50000 nM T13127 C6UA4Q 2819808 IC50 = 16000 nM T13127 C3H7IT 2826166 IC50 = 10 nM T13127 CNF42H 3005532 IC50 = 0.5 nM T13127 CNG05L 3012117 IC50 = 17 nM T13127 CQWM78 3350112 IC50 = 60 nM T13127 CPE3R7 3458143 IC50 = 3560 nM T13127 CO09CR 3481678 IC50 = 0.38 nM T13127 CF8NC7 3768552 IC50 > 1000000 nM T13127 CHAE56 4369208 IC50 = 37 nM T13127 CZ1WD3 4476323 IC50 = 59000 nM T13127 C9ZMC4 4476324 IC50 = 59000 nM T13127 C9XUM2 4631604 IC50 = 2.2 nM T13127 CI0MO5 5255691 IC50 = 30300 nM T13127 CGI02W 5287820 IC50 = 0.06 nM T13127 C2SVG1 5288261 IC50 = 130 nM T13127 C8EG4K 5326625 IC50 = 1.1 nM T13127 CYMQ90 5362708 IC50 > 1000000 nM T13127 CL5B2Z 5734804 IC50 = 8800 nM T13127 CR9N0A 6026467 IC50 = 402000 nM T13127 CJ9K4H 6041389 IC50 = 5140 nM T13127 CHG13F 6273500 IC50 = 11.9 nM T13127 C4IB9F 6504852 IC50 = 2580 nM T13127 C65LNA 6918349 IC50 = 350 nM T13127 C6GU9P 6918458 IC50 = 34000 nM T13127 CT7NM0 9499174 IC50 = 3220 nM T13127 CWKP41 9541655 IC50 = 3890 nM T13127 CDXJ85 9592460 IC50 = 51.5 nM T13127 CYB9H1 9796689 IC50 = 53 nM T13127 C8SGZ7 9799609 IC50 = 85 nM T13127 CZYW17 9801069 IC50 = 2.2 nM T13127 C0DXP2 9802891 IC50 = 9200 nM T13127 C90ETG 9803411 IC50 = 1.9 nM T13127 CK6GL7 9803684 IC50 = 1520 nM T13127 CZ8X4D 9803863 IC50 = 14 nM T13127 C5FKO9 9804240 IC50 = 102 nM T13127 CI29LC 9804512 IC50 = 11 nM T13127 C90GKJ 9804961 IC50 = 30 nM T13127 CN4Q9X 9805861 IC50 = 155 nM T13127 CP3Z2Q 9805897 IC50 = 9 nM T13127 CN20EG 9805907 IC50 = 7 nM T13127 C2H4ZK 9806118 IC50 = 15 nM T13127 C2TN7S 9807068 IC50 = 6.1 nM T13127 CWEC47 9807535 IC50 = 13 nM T13127 CC0F8G 9809539 IC50 = 5 nM T13127 CPZR70 9809959 IC50 = 0.4 nM T13127 CK5H4S 9810043 IC50 = 260 nM T13127 C8NXK4 9810235 IC50 = 2.1 nM T13127 CWCU84 9810607 IC50 = 76.1 nM T13127 CG53ZB 9819469 IC50 = 41500 nM T13127 CQD29O 9820245 IC50 < 1 nM T13127 C71XRT 9821510 IC50 = 5.7 nM T13127 C7LJV0 9823033 IC50 = 20000 nM T13127 C6R3OZ 9823857 IC50 = 36 nM T13127 CIE8J3 9823960 IC50 = 34 nM T13127 CEL3C9 9824630 IC50 = 17 nM T13127 CR9KA6 9825413 IC50 = 517 nM T13127 C2UCQ0 9825504 IC50 = 5 nM T13127 C6OR1H 9827026 IC50 = 99 nM T13127 C2A1DT 9827175 IC50 = 920 nM T13127 C2CVQ8 9828040 IC50 = 0.9 nM T13127 CQ0S9K 9828127 IC50 = 1.1 nM T13127 CI6N9C 9828259 IC50 = 2000 nM T13127 C5W3HI 9829059 IC50 = 1600 nM T13127 CUFZ58 9830366 IC50 = 42 nM T13127 CY3QP4 9830999 IC50 = 2.1 nM T13127 CB1CL6 9831259 IC50 = 2 nM T13127 CPX94T 9831633 IC50 = 4.3 nM T13127 CD39TX 9831734 IC50 = 5.3 nM T13127 C17VHW 9841030 IC50 = 123 nM T13127 CCY0V2 9842387 IC50 = 72 nM T13127 CXE1Y8 9842436 IC50 = 43 nM T13127 CA6N0H 9843867 EC50 = 6.1 nM T13127 CISP20 9844227 IC50 = 21 nM T13127 CE1BV0 9844383 IC50 = 4.3 nM T13127 C9EF7P 9844957 IC50 = 460 nM T13127 CD8R0L 9845012 IC50 = 11000 nM T13127 CNE6P0 9845017 IC50 = 2.7 nM T13127 C7VSU2 9845018 IC50 = 1.9 nM T13127 CXH80T 9845019 IC50 = 25 nM T13127 C41MGE 9845469 IC50 = 0.95 nM T13127 C8OFP0 9845527 IC50 = 19 nM T13127 CNIS42 9846821 IC50 = 0.4 nM T13127 CU3W1A 9846868 IC50 = 5400 nM T13127 CQ71HF 9847434 IC50 = 1790 nM T13127 CNC27L 9848289 IC50 = 43 nM T13127 C57GKV 9848392 IC50 = 891.25 nM T13127 CML5U3 9848397 IC50 = 51 nM T13127 C04ZEC 9848802 IC50 = 2.6 nM T13127 CSRA08 9848861 IC50 = 0.6 nM T13127 C4HSF1 9849786 IC50 = 110 nM T13127 C5L7CZ 9850092 IC50 = 3.6 nM T13127 CGJ3Y2 9850193 IC50 = 20 nM T13127 C5XU7Q 9852718 IC50 = 2.6 nM T13127 CGV0N3 9852766 IC50 = 2.7 nM T13127 CDX63H 9853141 IC50 = 7.8 nM T13127 C51YZX 9860658 IC50 = 3500 nM T13127 CT3CW6 9862094 IC50 = 1.1 nM T13127 C3ED5W 9862427 IC50 = 40 nM T13127 CAT1P0 9862539 IC50 = 1 nM T13127 C0AD8N 9863840 IC50 = 5 nM T13127 C81UHJ 9866014 IC50 = 100000 nM T13127 CYH4A5 9866559 IC50 = 183 nM T13127 CXZ6Q7 9866918 IC50 = 9.5 nM T13127 C24VHZ 9866971 IC50 = 4.5 nM T13127 CAOK24 9867098 IC50 < 1 nM T13127 C9RJQ8 9867301 IC50 = 62.9 nM T13127 CJE1C8 9867500 IC50 = 140 nM T13127 CND3X4 9868632 IC50 = 0.44 nM T13127 CDG2H9 9868693 IC50 = 2600 nM T13127 CZ7S2M 9869309 EC50 = 0.5 nM T13127 CUE43P 9869839 EC50 = 3.5 nM T13127 CQNZ19 9870627 IC50 = 0.5 nM T13127 C4K3AC 9870962 IC50 = 5.7 nM T13127 CWD56L 9871581 IC50 = 11 nM T13127 C0QV1K 9871743 IC50 = 6 nM T13127 CR6SP4 9872991 IC50 = 310 nM T13127 CZN6S0 9873563 IC50 = 3.9 nM T13127 CCXO64 9873605 IC50 = 62 nM T13127 CF0B4E 9874946 IC50 < 10 nM T13127 CQ87TL 9875356 IC50 = 17.1 nM T13127 C4NJS0 9885760 IC50 = 200 nM T13127 CS8GL2 9886161 IC50 = 160 nM T13127 CD8F7K 9887967 IC50 = 8 nM T13127 C7YD9E 9888084 IC50 = 21.8 nM T13127 CF80UP 9889061 IC50 = 14 nM T13127 CM5GI2 9889827 IC50 = 54 nM T13127 CSR2H6 9889842 IC50 = 4200 nM T13127 CV97PM 9890363 IC50 = 0.2 nM T13127 C9DYL4 9890611 IC50 = 520 nM T13127 CCA2R6 9891061 IC50 = 7000 nM T13127 C4MPO6 9891092 IC50 = 1 nM T13127 CC36ED 9891239 IC50 = 1.1 nM T13127 CN31TA 9891465 IC50 = 59 nM T13127 CO6AF7 9891655 IC50 = 4 nM T13127 C4D5NZ 9891739 IC50 = 1.7 nM T13127 CM0JO5 9891920 Ki = 4.5 nM T13127 CU1FV4 9892151 IC50 = 0.47 nM T13127 C15RFY 9892214 IC50 = 7.4 nM T13127 CW64AK 9894120 IC50 = 1000 nM T13127 CPR23Q 9896461 IC50 = 4.3 nM T13127 CRW8C1 9907452 IC50 = 27 nM T13127 CU0NJ8 9910183 IC50 = 11 nM T13127 CB87AX 9912725 IC50 = 1.13 nM T13127 CA8KC0 9912881 IC50 = 7.5 nM T13127 CNG36R 9913024 IC50 = 560 nM T13127 CH4SI7 9913660 IC50 = 3.5 nM T13127 CW1KP6 9914569 IC50 = 42 nM T13127 CHQC65 9914869 IC50 = 47 nM T13127 CF85LV 9915185 IC50 = 2.5 nM T13127 C4KG9M 9916011 EC50 = 28 nM T13127 C9YUE6 9917374 IC50 = 78 nM T13127 C69MCF 9930166 IC50 = 3 nM T13127 CH2KA7 9930818 IC50 = 230 nM T13127 CY7W8H 9931146 IC50 = 1.5 nM T13127 CM6PZ0 9931933 IC50 = 1000 nM T13127 CJ93FZ 9932066 IC50 = 1.3 nM T13127 C9FZO7 9932679 IC50 = 3.5 nM T13127 C8QKA9 9932796 IC50 = 8.4 nM T13127 C5HQM7 9932974 EC50 = 0.12 nM T13127 C5OU0K 9933592 IC50 = 1.4 nM T13127 C2YR7H 9933648 IC50 = 590 nM T13127 C8RG7D 9933894 IC50 = 10.9 nM T13127 CHFS82 9933907 IC50 = 4.52 nM T13127 CA3C4E 9933908 IC50 = 0.48 nM T13127 C2YJL6 9934578 IC50 = 3 nM T13127 CW17BV 9935094 IC50 = 74 nM T13127 C4YUR9 9935680 IC50 = 2.2 nM T13127 CI9D2M 9935716 IC50 = 3.5 nM T13127 CN9HX5 9936941 IC50 = 310 nM T13127 CQ7D1C 9937451 IC50 = 38 nM T13127 C9R0FV 9938283 IC50 = 10000 nM T13127 CYX02E 9938720 IC50 = 850 nM T13127 C5C2NJ 9939360 IC50 = 170 nM T13127 C84CME 9939472 IC50 = 1.9 nM T13127 C4SBH7 9947735 IC50 = 8641 nM T13127 CI8P9X 9952087 IC50 = 21 nM T13127 C9HB0W 9952272 IC50 = 1900 nM T13127 C5PK0N 9952667 EC50 = 1000 nM T13127 C2U8FH 9954480 IC50 = 160 nM T13127 C4LJC2 9954534 IC50 = 500 nM T13127 C3MSB4 9954645 IC50 = 0.1 nM T13127 C9V3EF 9955169 IC50 = 3.1 nM T13127 C8TB6H 9955707 IC50 = 8000 nM T13127 C6RC0B 9956145 IC50 = 200 nM T13127 CW71XF 9956883 IC50 = 19 nM T13127 CNRX39 9956928 EC50 = 3.86 nM T13127 CJ5QB9 9957218 IC50 = 6.5 nM T13127 C3D8SE 9957733 IC50 = 38 nM T13127 CSR1X7 9958087 IC50 = 0.33 nM T13127 C3HC2Z 9958709 IC50 = 41 nM T13127 C6R0FK 9959504 IC50 = 49 nM T13127 C9A1HU 9960439 IC50 = 2.6 nM T13127 CT6Q7F 9961463 IC50 = 3.1 nM T13127 CSKW34 9968685 IC50 = 712 nM T13127 C38VQR 9969350 IC50 = 43 nM T13127 CH9R1L 9972169 IC50 = 543 nM T13127 C4HL7Q 9981319 IC50 = 1 nM T13127 CBFW98 9982211 IC50 = 1.4 nM T13127 CM65XN 10022561 IC50 = 20 nM T13127 C9RGX6 10022869 IC50 = 1900 nM T13127 C3DGR5 10024805 IC50 = 3.3 nM T13127 CC90RP 10024865 IC50 = 17750 nM T13127 C2EA8Y 10025359 IC50 = 31 nM T13127 C7MBZ0 10026704 IC50 = 740 nM T13127 C3AK9T 10043886 IC50 = 4600 nM T13127 CMCB24 10046604 IC50 = 1700 nM T13127 CESP05 10049294 IC50 = 8 nM T13127 C1LHE6 10050983 IC50 = 1.77 nM T13127 CG8K9B 10051380 IC50 = 24 nM T13127 CF93OV 10052548 IC50 = 52 nM T13127 CQPF91 10054901 IC50 = 2.5 nM T13127 CQ85UN 10067611 IC50 = 15000 nM T13127 C0XTN6 10070247 IC50 = 2400 nM T13127 CCU3L2 10072355 IC50 = 130 nM T13127 CCBL59 10072414 IC50 = 1.77 nM T13127 C61SKV 10078035 IC50 = 330 nM T13127 CTP3V8 10078563 IC50 = 2.1 nM T13127 C2JO1F 10090255 IC50 = 30000 nM T13127 CU4ZN5 10091605 IC50 = 250 nM T13127 C67SBQ 10092425 IC50 = 1000 nM T13127 CF4KW7 10093287 IC50 = 530 nM T13127 CO1Y0A 10094096 IC50 = 13000 nM T13127 CJR8C6 10096236 IC50 = 3000 nM T13127 CFWY79 10099159 IC50 = 3400 nM T13127 CQW6T2 10101158 IC50 = 400 nM T13127 C1B2XO 10102159 IC50 = 145 nM T13127 C0V8RA 10108995 IC50 = 182 nM T13127 CI1KL0 10113666 IC50 = 2733 nM T13127 C3AI1G 10114664 EC50 = 525 nM T13127 CAPF20 10116169 EC50 = 7.3 nM T13127 CC5NS4 10116426 IC50 = 2150 nM T13127 CI06LE 10116437 IC50 = 5 nM T13127 CCFE56 10117200 IC50 = 5 nM T13127 CY41IQ 10117731 IC50 = 17 nM T13127 CXK1F5 10121539 IC50 = 311 nM T13127 CF0U6B 10122788 IC50 = 25 nM T13127 CV35EA 10127337 EC50 = 5.2 nM T13127 C05SCV 10135324 IC50 = 44 nM T13127 CL4VY5 10137458 IC50 = 800 nM T13127 CE9OF2 10138363 EC50 = 100 nM T13127 CT9F1M 10138638 EC50 = 390 nM T13127 C83ZYO 10138658 EC50 < 1 nM T13127 CTL6F2 10140413 IC50 = 572 nM T13127 C1H8TO 10142164 IC50 = 0.9 nM T13127 CX42MQ 10143267 IC50 = 350 nM T13127 C39ZKT 10146069 IC50 = 2000 nM T13127 C1OTC6 10156140 IC50 = 241 nM T13127 CGT8Y1 10156869 IC50 = 232 nM T13127 CI63TS 10156870 IC50 = 400 nM T13127 CJ2Q1T 10156985 IC50 = 245 nM T13127 CE7C2O 10157539 IC50 = 160 nM T13127 CAU31X 10157671 IC50 = 8685 nM T13127 C4FPQ9 10157672 IC50 = 1500 nM T13127 C4FXS8 10157673 IC50 = 2484 nM T13127 C1YVE7 10158436 IC50 = 11389 nM T13127 CW0Z5M 10158556 IC50 = 3803 nM T13127 CW98LU 10162566 IC50 = 54 nM T13127 CRIA34 10163807 EC50 = 13 nM T13127 CZ2KM3 10164142 IC50 = 1.6 nM T13127 C0YU2R 10177303 IC50 = 110 nM T13127 C7M5QO 10177652 IC50 = 1628 nM T13127 C9XTL1 10177877 IC50 = 171 nM T13127 CMJ4R0 10178945 IC50 = 4588 nM T13127 CV3W0U 10179853 IC50 = 12 nM T13127 C26CJM 10180787 IC50 = 29863 nM T13127 C5QL4V 10182213 IC50 = 19 nM T13127 CDR9T1 10182250 EC50 > 1000 nM T13127 COKV74 10185561 IC50 = 0.46 nM T13127 CWOB16 10187763 IC50 = 8 nM T13127 CTRQ41 10195107 EC50 = 0.19 nM T13127 C53ZSL 10195730 IC50 = 1.4 nM T13127 CYNZ58 10199980 IC50 = 684 nM T13127 CNAS15 10201818 IC50 = 1372 nM T13127 CQY5F9 10204944 IC50 = 14369 nM T13127 C5JW6T 10207204 IC50 = 1.2 nM T13127 C2YEM7 10212166 IC50 = 360 nM T13127 C9I4QZ 10221771 IC50 = 568 nM T13127 CYX25D 10223743 IC50 = 46 nM T13127 CRUY32 10226337 EC50 = 4.6 nM T13127 CBW57M 10233954 IC50 = 2 nM T13127 C5BJ0E 10238214 EC50 = 0.75 nM T13127 CE34HG 10253040 EC50 = 12 nM T13127 CXN63O 10253506 IC50 > 10000 nM T13127 CWS7U0 10253637 IC50 = 95000 nM T13127 CY4GO6 10256312 IC50 = 31 nM T13127 C7NR8Z 10271199 IC50 = 45 nM T13127 C2AS9M 10271497 IC50 = 527 nM T13127 C0WL3V 10272144 IC50 = 3900 nM T13127 C2U5PZ 10272943 IC50 = 4004 nM T13127 CPSF82 10273485 IC50 = 172 nM T13127 CQC6U4 10277213 IC50 = 1740 nM T13127 C9EUI2 10278364 IC50 = 5.5 nM T13127 CQK7V3 10278841 IC50 = 0.97 nM T13127 CX49UK 10279599 EC50 = 3.9 nM T13127 CI0LU5 10279755 IC50 = 29 nM T13127 C19YTB 10280112 IC50 = 93 nM T13127 C1R8UJ 10288135 IC50 = 2500 nM T13127 C83BMF 10293350 IC50 = 58 nM T13127 C6CTB5 10294243 IC50 = 77 nM T13127 C02NRB 10300220 IC50 = 2.2 nM T13127 CP8M7E 10311107 IC50 = 6.4 nM T13127 CVA36C 10319260 IC50 = 18 nM T13127 CR5O7S 10319572 IC50 = 1 nM T13127 C2KAT9 10320387 IC50 = 2.9 nM T13127 C1MD0E 10321796 IC50 = 19700 nM T13127 CO31ND 10341436 IC50 = 700 nM T13127 C09KJE 10342485 IC50 = 8700 nM T13127 CM8OQ2 10343264 IC50 = 20 nM T13127 C1QIA6 10346600 IC50 = 480 nM T13127 CQN71K 10348643 IC50 = 40 nM T13127 CGU61W 10349177 IC50 > 280 nM T13127 CR5AN4 10349221 IC50 = 1.7 nM T13127 CZ8F6U 10350609 IC50 = 3990 nM T13127 C4BL0X 10358625 IC50 = 40000 nM T13127 CJWK53 10362198 IC50 > 1000000 nM T13127 C1I3CY 10366632 IC50 = 930 nM T13127 CP31VA 10367960 IC50 = 820 nM T13127 CKV30M 10368622 IC50 = 660 nM T13127 COTF69 10368623 IC50 = 110 nM T13127 CS3Q2L 10368640 IC50 = 380 nM T13127 CPY2W3 10369223 IC50 = 0.92 nM T13127 CP1X4H 10369934 IC50 = 10.6 nM T13127 C13IDM 10371139 IC50 = 250 nM T13127 CB25TJ 10371983 IC50 = 60 nM T13127 CE9I4H 10386837 IC50 = 35 nM T13127 CZ6XN0 10387250 IC50 = 55000 nM T13127 C7XOR8 10387426 IC50 = 5600 nM T13127 C4MXB5 10389076 IC50 = 0.4 nM T13127 C8YOX7 10389736 IC50 = 1000 nM T13127 CP0CA7 10390566 IC50 = 4.6 nM T13127 C0AK8P 10390583 IC50 = 26 nM T13127 C3DN4J 10390776 IC50 = 0.62 nM T13127 C3YE9J 10393519 IC50 = 3500 nM T13127 CE08BL 10402973 IC50 = 115000 nM T13127 CCA9P1 10403581 IC50 = 748000 nM T13127 CB3E0V 10403878 IC50 = 130000 nM T13127 CO82YZ 10404984 IC50 > 30000 nM T13127 C5UJ4I 10407776 IC50 = 5400 nM T13127 C4K9FO 10408744 IC50 = 50 nM T13127 CCH02G 10410157 IC50 > 10000 nM T13127 CBEZ75 10413692 IC50 = 0.79 nM T13127 CK8FQ5 10414268 IC50 = 310 nM T13127 CX0V4N 10416697 IC50 > 94 nM T13127 CH6NM2 10431162 IC50 = 75 nM T13127 CAF5X3 10432980 IC50 = 530 nM T13127 CY8P1G 10438437 IC50 = 0.41 nM T13127 CR2UK0 10448769 IC50 = 220000 nM T13127 C3U5MK 10450596 IC50 = 12600 nM T13127 C4QE3X 10450992 IC50 = 150 nM T13127 C32ZWY 10454373 IC50 = 22200 nM T13127 CT65RW 10455264 IC50 = 560000 nM T13127 CW03VF 10456723 IC50 = 1300 nM T13127 C6UY4R 10458946 IC50 = 60 nM T13127 CSD3H4 10461317 IC50 = 5 nM T13127 C61CXN 10461791 IC50 = 3.1 nM T13127 CY93IH 10473146 IC50 = 25000 nM T13127 CXW9P3 10474028 IC50 = 11500 nM T13127 CR6J8W 10478749 IC50 = 0.61 nM T13127 CIS0C3 10478862 IC50 = 1170 nM T13127 C6XTW8 10484625 IC50 = 6.2 nM T13127 CUR59W 10496660 IC50 = 100000 nM T13127 CR8D7M 10497786 IC50 = 13600 nM T13127 C2I0XQ 10500948 IC50 = 1100 nM T13127 CY0SD2 10501521 IC50 = 10000 nM T13127 CMN38Y 10501927 IC50 = 17 nM T13127 CK9DL0 10502155 IC50 = 23000 nM T13127 CRO4G8 10503666 IC50 = 2300 nM T13127 C3J4UD 10503667 IC50 = 910 nM T13127 CTM2A7 10503879 IC50 = 470 nM T13127 CHU7L9 10504242 IC50 = 0.11 nM T13127 CBGX73 10504791 IC50 = 2200 nM T13127 CP8WY6 10504845 IC50 = 1.53 nM T13127 C24OTY 10504924 IC50 = 3100 nM T13127 CRF2C7 10506309 IC50 = 40 nM T13127 CA43JZ 10506447 IC50 = 41 nM T13127 CZOH48 10506589 IC50 = 7400 nM T13127 CWI8Z5 10507119 IC50 = 6 nM T13127 CW52BG 10507372 IC50 = 50 nM T13127 CFY47V 10507892 IC50 = 2.3 nM T13127 C8F7PV 10508462 IC50 > 360000 nM T13127 CZ43JV 10519494 IC50 = 11000 nM T13127 C83LTO 10523971 IC50 = 21000 nM T13127 C2QDH7 10524137 IC50 = 8.75 nM T13127 C1V2KO 10524482 IC50 = 1300 nM T13127 CW0M9U 10525430 IC50 = 25800 nM T13127 C2WDZ5 10526212 IC50 = 48 nM T13127 C28VQG 10526694 IC50 = 1600 nM T13127 CRV3F2 10527488 IC50 = 490 nM T13127 CRW9O0 10527651 IC50 = 600 nM T13127 CW41MH 10527921 IC50 = 15400 nM T13127 CN06HX 10528235 IC50 = 4100 nM T13127 C7RT4O 10528378 IC50 = 4800 nM T13127 C4U9EY 10528921 IC50 > 4000 nM T13127 C8UF6E 10528967 IC50 = 1000 nM T13127 CD5UM0 10529689 IC50 = 24 nM T13127 CS9HN0 10529690 IC50 = 18 nM T13127 CS9M5T 10529724 IC50 = 5100 nM T13127 CP4D7J 10530034 IC50 = 35500 nM T13127 C4L2YP 10530192 IC50 = 400 nM T13127 CA4V2K 10530612 IC50 = 86 nM T13127 CEC5U4 10549323 IC50 = 34000 nM T13127 C23XOP 10549461 IC50 = 700 nM T13127 CZCE90 10549651 IC50 = 1500 nM T13127 CSC2Y4 10549858 IC50 = 540000 nM T13127 CNA5R7 10549950 IC50 = 480 nM T13127 C74EOD 10550035 IC50 = 9 nM T13127 C7D6CO 10550114 IC50 = 3 nM T13127 CE6G2U 10550323 IC50 = 5400 nM T13127 C56SID 10550324 IC50 = 1200 nM T13127 C6UEY5 10550770 IC50 = 900 nM T13127 CV48DZ 10550827 IC50 = 500 nM T13127 CEQ76B 10551282 IC50 = 2968000 nM T13127 C1UG5S 10551942 IC50 = 850 nM T13127 C4JOR7 10552209 IC50 = 100000 nM T13127 C3J2SP 10552253 IC50 = 15000 nM T13127 CO28TX 10552504 IC50 = 10.7 nM T13127 CGYL12 10552882 IC50 = 124000 nM T13127 CRA56B 10553781 IC50 = 12 nM T13127 CJH3P9 10553926 IC50 = 87 nM T13127 CK1SC0 10554866 IC50 = 45 nM T13127 CNJ3M4 10554914 IC50 > 110 nM T13127 C0SBQ7 10555567 IC50 = 1400 nM T13127 CZ93OG 10566622 IC50 = 8500 nM T13127 CDS0I5 10573470 IC50 = 9800 nM T13127 CT0UH4 10574311 IC50 = 4.8 nM T13127 C0PUZ4 10574391 IC50 > 10000 nM T13127 CT12WR 10574411 IC50 = 1400 nM T13127 C3WJ5I 10574866 IC50 = 1280 nM T13127 CI79WP 10575347 IC50 = 530 nM T13127 C0UAF6 10575390 IC50 = 4900 nM T13127 CS0T9C 10575431 IC50 = 650 nM T13127 C6NIT3 10575560 IC50 = 2.85 nM T13127 CV67HL 10575577 IC50 = 1370 nM T13127 CZ03TM 10576001 IC50 = 715 nM T13127 CUP42G 10576440 IC50 = 383 nM T13127 CKB80J 10576441 IC50 = 5.95 nM T13127 CQ7CI5 10576442 IC50 = 7.9 nM T13127 CD9L6W 10576892 IC50 = 2500 nM T13127 CPF43H 10577225 IC50 = 7000 nM T13127 CF9O8Z 10578069 IC50 = 500 nM T13127 CI4DU3 10578336 IC50 = 12200 nM T13127 C7JUZ5 10591506 IC50 = 13500 nM T13127 CTQW71 10597499 IC50 = 48000 nM T13127 CS2XG1 10597618 IC50 = 4400 nM T13127 CX2W8Z 10598227 IC50 = 27000 nM T13127 CFNX62 10598287 IC50 = 325 nM T13127 C45PUT 10598485 IC50 = 200 nM T13127 CKU61I 10598920 IC50 = 800 nM T13127 CG5S2F 10599760 IC50 = 1190 nM T13127 CRN17G 10600336 IC50 = 58000 nM T13127 CWJ6N9 10600539 IC50 = 1300 nM T13127 CIO94A 10601507 IC50 = 28500 nM T13127 CQV3G0 10601641 IC50 = 101 nM T13127 CE41UR 10601829 IC50 = 880 nM T13127 C05YMT 10601986 IC50 = 86 nM T13127 CT74GP 10602162 IC50 = 30 nM T13127 C1VW2I 10602521 IC50 = 900 nM T13127 C45DSZ 10602865 IC50 = 68 nM T13127 C9EZ8C 10603585 IC50 = 45000 nM T13127 CX8D6R 10614321 IC50 = 4575 nM T13127 CSG8O6 10619608 IC50 = 3800 nM T13127 C03FOD 10620775 IC50 = 350000 nM T13127 CUS69I 10622279 IC50 = 11300 nM T13127 CT0MP2 10622831 IC50 = 600 nM T13127 CD48WE 10623317 IC50 = 3800 nM T13127 C7V4ID 10623379 IC50 = 7000 nM T13127 C1D7MR 10623537 IC50 = 700 nM T13127 C0X5HL 10624014 IC50 = 186000 nM T13127 CBW58Q 10624371 IC50 = 437 nM T13127 C50TNK 10625063 IC50 = 1050 nM T13127 CZ0D4E 10625093 IC50 = 0.6 nM T13127 CSX5T2 10625933 IC50 = 1100 nM T13127 C65KOH 10626112 IC50 = 54 nM T13127 C0XYW2 10626134 IC50 = 300 nM T13127 CO0U1T 10626514 IC50 > 360000 nM T13127 CMGH39 10626729 IC50 < 3.8 nM T13127 CBD5S0 10627659 IC50 = 1700 nM T13127 CU1S2T 10644481 IC50 = 1300 nM T13127 C8AD9L 10644482 IC50 = 2000 nM T13127 CF9M3D 10645020 IC50 = 1300 nM T13127 C3NTM0 10645959 IC50 = 1200 nM T13127 C3F1MQ 10646360 IC50 = 2730 nM T13127 C01DPW 10646414 IC50 = 1090 nM T13127 CFQ5A4 10647085 IC50 = 2000 nM T13127 CEZ32R 10647125 IC50 = 4600 nM T13127 CU15YE 10647606 IC50 = 177000 nM T13127 C9A3HI 10647676 IC50 = 1740 nM T13127 C7SH8F 10647793 IC50 = 205000 nM T13127 CUE30Q 10648132 IC50 = 276 nM T13127 CCYK64 10648442 IC50 = 23.5 nM T13127 C85KQP 10648955 IC50 = 1300 nM T13127 CO6XV1 10649291 IC50 = 18100 nM T13127 CW9MZ2 10649434 IC50 = 210 nM T13127 C9P4XE 10649859 IC50 = 3600 nM T13127 C2D8KM 10650059 IC50 = 249000 nM T13127 C0ZTV9 10650576 IC50 = 38000 nM T13127 C42BIA 10650822 IC50 = 69 nM T13127 C1R2NH 10651878 IC50 = 5.3 nM T13127 CEW31H 10652422 IC50 = 2.5 nM T13127 CF3PT6 10665097 IC50 = 32000 nM T13127 CC8Q7I 10669102 IC50 = 38300 nM T13127 CZ01XM 10670109 IC50 = 720 nM T13127 C1P3JX 10670356 IC50 = 880 nM T13127 CMN93V 10670701 IC50 = 1250 nM T13127 C9VRT5 10671919 IC50 = 1270 nM T13127 C34FCV 10672663 IC50 = 54.5 nM T13127 C3QBU9 10674120 IC50 = 33.1 nM T13127 C2MD9S 10674325 IC50 = 380 nM T13127 C07EIR 10675788 IC50 = 30500 nM T13127 CN9KY1 10691938 IC50 = 2300 nM T13127 CMC15X 10693478 IC50 = 303 nM T13127 C5Y2LS 10693493 IC50 = 210 nM T13127 CB4J2E 10694111 IC50 = 950 nM T13127 CV0CZ3 10694627 IC50 = 1000 nM T13127 CSKZ49 10694662 IC50 = 640 nM T13127 C1HZ0C 10694872 IC50 = 3100 nM T13127 CG38AJ 10695790 IC50 = 54.5 nM T13127 C2VJF6 10696114 IC50 = 1600 nM T13127 C5VF3S 10696316 IC50 = 1770 nM T13127 CIJO54 10697049 IC50 = 2900 nM T13127 C69VAQ 10697182 IC50 = 83 nM T13127 C64IKV 10697405 IC50 = 20000 nM T13127 CDX93R 10697659 IC50 = 1000 nM T13127 CSRP16 10698121 IC50 = 43 nM T13127 CJTP72 10698563 IC50 < 250 nM T13127 CR4H9W 10715827 IC50 = 1000000 nM T13127 CS5IF2 10716401 IC50 = 320 nM T13127 COMP10 10717281 IC50 = 1300 nM T13127 CGU3D7 10717672 IC50 = 3200 nM T13127 CQ2IU7 10717718 IC50 = 820 nM T13127 C56SFP 10717901 IC50 = 60 nM T13127 CI4KE6 10718316 IC50 = 702000 nM T13127 C1LC3H 10718487 IC50 = 640 nM T13127 C40WHQ 10718836 IC50 > 360000 nM T13127 C4UB8M 10719050 IC50 = 4300 nM T13127 C3SK7O 10719054 IC50 = 880 nM T13127 CA6OI7 10719279 IC50 = 16 nM T13127 C9HLF4 10719575 IC50 = 19000 nM T13127 C2LBA4 10719577 IC50 = 1750 nM T13127 CR32TN 10719770 IC50 = 114 nM T13127 CG0FQ7 10719802 IC50 = 58000 nM T13127 C41TBI 10720216 IC50 = 820 nM T13127 CT3AO5 10720557 IC50 = 4800 nM T13127 CCE4Z2 10720963 IC50 = 280 nM T13127 CG2JH6 10721003 IC50 = 54 nM T13127 CT1DJ5 10721277 IC50 = 16.7 nM T13127 CUAN03 10721615 IC50 > 360000 nM T13127 CE4P6G 10729939 IC50 = 1070 nM T13127 C28OAJ 10730506 IC50 > 75000 nM T13127 C0KW4X 10730919 IC50 = 710 nM T13127 CWH73L 10734205 IC50 = 917 nM T13127 CI2M1J 10737397 IC50 = 1100 nM T13127 CO1C9D 10739566 IC50 = 2500 nM T13127 CW0A3Q 10741064 IC50 = 5300 nM T13127 CH7FU9 10742050 IC50 = 4500 nM T13127 CRBZ62 10742589 IC50 = 145000 nM T13127 C8DIN9 10742774 IC50 = 72 nM T13127 C5V9AT 10743067 IC50 = 1100 nM T13127 CJ6AR0 10743164 IC50 = 2440 nM T13127 CD2Y5W 10743390 IC50 = 1423000 nM T13127 C07AMC 10743633 IC50 = 45 nM T13127 C7F0QS 10744252 IC50 = 160 nM T13127 CZ6GT5 10744467 IC50 = 78 nM T13127 C1BWA8 10744607 IC50 = 880 nM T13127 CX95GM 10744748 IC50 = 210 nM T13127 CIW3K0 10745350 IC50 = 5000 nM T13127 CZSF85 10745444 IC50 = 102 nM T13127 CRB58V 10746457 IC50 = 230 nM T13127 C5YQV8 10752959 IC50 = 266000 nM T13127 C4R1UI 10763925 IC50 = 5.6 nM T13127 C34CRF 10763992 IC50 = 2700 nM T13127 CR2MU7 10764061 IC50 = 590 nM T13127 C6H4MZ 10764416 IC50 = 10800 nM T13127 CFL49O 10765113 IC50 = 10700 nM T13127 CTRO45 10765213 IC50 = 190 nM T13127 C6YCJ3 10765492 IC50 = 1100 nM T13127 C5KO9X 10765627 IC50 = 1100 nM T13127 C74ZJY 10765816 IC50 = 4100 nM T13127 C2XYA0 10765908 IC50 = 1200 nM T13127 C4Q3HS 10765989 IC50 = 1660 nM T13127 CTN7O5 10766165 IC50 = 2100 nM T13127 CQ9K2I 10766334 IC50 = 2780 nM T13127 C0SAR8 10766655 IC50 = 1800 nM T13127 C9J8WF 10767556 IC50 = 2100 nM T13127 C2P4OA 10767597 IC50 = 13300 nM T13127 CTKI31 10768220 IC50 = 170 nM T13127 C0I5XK 10768364 IC50 = 4600 nM T13127 C05RKS 10768376 IC50 = 28000 nM T13127 C20WCZ 10768592 IC50 = 450 nM T13127 CZ7G8E 10769617 IC50 = 60 nM T13127 CZP71M 10769930 IC50 = 100 nM T13127 C9YH6Q 10769977 IC50 = 2 nM T13127 CIX79V 10770123 IC50 = 27 nM T13127 CIL16U 10786579 IC50 = 44 nM T13127 CZH9O0 10786711 IC50 = 3200 nM T13127 CHS34P 10786765 IC50 = 2570 nM T13127 C7FA5Y 10786932 IC50 = 340 nM T13127 CNS05M 10787875 IC50 = 20800 nM T13127 CK4E2G 10788891 IC50 = 360 nM T13127 CWS20Y 10789192 IC50 = 168000 nM T13127 CB3I0A 10789410 IC50 = 550 nM T13127 CX21PO 10789480 IC50 = 2600 nM T13127 CQ2W9M 10789829 IC50 = 1800 nM T13127 CH46CT 10790170 IC50 = 228 nM T13127 CI2JV3 10790910 IC50 = 870 nM T13127 C9L1XH 10790911 IC50 = 3500 nM T13127 C3QK4D 10791550 IC50 = 84 nM T13127 CN38DU 10791803 IC50 = 2500 nM T13127 CKI5J3 10792917 IC50 = 23000 nM T13127 C8SOF1 10792989 IC50 = 48 nM T13127 CT1H0F 10793775 IC50 > 95 nM T13127 CQT9B6 10794150 IC50 = 42500 nM T13127 C4B1YP 10796012 IC50 = 20 nM T13127 C9GV2H 10803148 IC50 > 70000 nM T13127 C8YS4A 10808491 IC50 = 1300 nM T13127 CAIR64 10808673 IC50 = 16000 nM T13127 CM1W7R 10809672 IC50 = 1300 nM T13127 C3L9PC 10811325 IC50 = 46000 nM T13127 CI97PH 10811576 IC50 = 840 nM T13127 C1NME7 10811789 IC50 = 22 nM T13127 CTB5P7 10812135 IC50 = 1250 nM T13127 C0Y3OQ 10812712 IC50 = 7300 nM T13127 C97OTM 10812928 IC50 = 700 nM T13127 C3QIN8 10812949 IC50 = 6800 nM T13127 CWS08X 10813620 IC50 = 35000 nM T13127 CGN4L2 10813810 IC50 = 3300 nM T13127 CP5OA8 10813811 IC50 = 12300 nM T13127 C45SWA 10814464 IC50 = 1260 nM T13127 C7E3UW 10814818 IC50 = 450 nM T13127 CY5G1Q 10815067 IC50 = 426000 nM T13127 CF67HY 10815603 IC50 = 170 nM T13127 CR9VW5 10816092 IC50 = 100 nM T13127 C42CJH 10816435 IC50 = 38000 nM T13127 C2MG6O 10816874 IC50 = 1890 nM T13127 CLO89V 10817478 IC50 = 3000 nM T13127 C1MXB5 10818167 IC50 = 5600 nM T13127 CS2W0T 10818818 IC50 = 2.2 nM T13127 C6SO2W 10818824 IC50 = 0.8 nM T13127 CH43SG 10833680 IC50 = 1800 nM T13127 CNW4H9 10834603 IC50 = 6000 nM T13127 CM40US 10836459 IC50 = 2500 nM T13127 C2JEN7 10837238 IC50 = 1800 nM T13127 CIMA72 10837502 IC50 = 2300 nM T13127 CWY78O 10837636 IC50 = 490 nM T13127 C8L1JF 10837699 IC50 = 20200 nM T13127 CHY91F 10837874 IC50 = 3800 nM T13127 C6ARE0 10837934 IC50 = 91000 nM T13127 CR6D3F 10838529 IC50 = 330 nM T13127 CV1WE9 10839035 IC50 = 430 nM T13127 CI35QL 10839833 IC50 = 350 nM T13127 CJZ60V 10841523 IC50 = 1290 nM T13127 CL2ZN3 10841787 IC50 = 340 nM T13127 COJI94 10862667 IC50 = 2900 nM T13127 CQ9K5G 10862882 IC50 = 1.4 nM T13127 CE9QF4 10863673 IC50 = 1.2 nM T13127 CX3RT7 10874250 IC50 = 1.2 nM T13127 CUO8C4 10874725 IC50 = 0.3 nM T13127 C7JNV1 10883893 IC50 = 100 nM T13127 C6KW8J 10884405 IC50 = 1800 nM T13127 C1FQ2V 10884731 IC50 = 0.6 nM T13127 C1NP4F 10893758 IC50 = 41 nM T13127 C3SM0F 10894628 IC50 = 270 nM T13127 C4QZ2E 10895064 IC50 = 27 nM T13127 CLI84D 10895869 IC50 = 2.3 nM T13127 CX9QO1 10896013 EC50 = 11 nM T13127 C5L2FR 10896860 IC50 = 18 nM T13127 CAB0O8 10906012 IC50 = 44 nM T13127 C3T9CI 10916025 IC50 = 120 nM T13127 C3SQA5 10918896 IC50 = 1.1 nM T13127 CD10XK 10928028 IC50 = 3.6 nM T13127 CEC8P2 10928657 IC50 = 52500 nM T13127 CYJ0H9 10938254 IC50 = 980 nM T13127 CISW28 10938819 IC50 > 10000 nM T13127 CSP40W 10949255 IC50 = 173 nM T13127 CG34TZ 10949393 IC50 = 610 nM T13127 CR8NL2 10950878 IC50 = 52 nM T13127 CQ10EL 10951981 IC50 = 5.8 nM T13127 C7MJ3I 10960344 IC50 = 250 nM T13127 CL3A7F 10961614 IC50 = 43 nM T13127 CZXI06 10971008 IC50 > 10000 nM T13127 CSE3C1 10971210 IC50 > 10000 nM T13127 C3I6QA 10972793 IC50 = 2900 nM T13127 CAX04J 10982806 IC50 > 10000 nM T13127 CS1CI9 10982914 IC50 = 83 nM T13127 CIS36R 10993420 IC50 = 150 nM T13127 CE6XI4 10993905 IC50 = 54 nM T13127 CFO35V 10994871 IC50 > 190 nM T13127 CJI01L 11004204 IC50 = 380 nM T13127 CC9W2Q 11015477 IC50 = 5.3 nM T13127 CH2A4Z 11016041 EC50 = 6.9 nM T13127 C2T8WC 11016388 IC50 = 0.46 nM T13127 CF2VN6 11016692 EC50 = 11 nM T13127 COK91D 11025039 IC50 = 2300 nM T13127 C2BX4N 11025461 IC50 = 110 nM T13127 CTFJ03 11026293 IC50 > 10000 nM T13127 C1N5EF 11026589 IC50 = 4.9 nM T13127 C4RJQ3 11037090 IC50 = 1.3 nM T13127 CPXY41 11037188 IC50 = 70 nM T13127 C4NWP7 11038422 IC50 = 1 nM T13127 CKZP84 11048052 IC50 = 65 nM T13127 C4X9QO 11048592 IC50 = 41700 nM T13127 CB9L4M 11059764 IC50 = 7.6 nM T13127 CJQ7D3 11060155 EC50 = 4 nM T13127 CR9K5V 11069519 IC50 = 8.4 nM T13127 CEM1Q6 11071188 IC50 = 450 nM T13127 C7YT0Q 11076782 IC50 = 170000 nM T13127 CN6QM7 11080796 IC50 = 4.8 nM T13127 C16QXU 11081452 IC50 = 5600 nM T13127 CP05LR 11090660 IC50 = 61 nM T13127 CV73YG 11091386 IC50 = 11 nM T13127 C2FIS6 11091715 IC50 = 1800 nM T13127 CBY94W 11091976 IC50 = 67 nM T13127 C5AO4V 11092095 IC50 = 430 nM T13127 C9RCT4 11092749 IC50 = 0.19 nM T13127 CY0F2S 11101410 IC50 = 250 nM T13127 C9COS1 11101729 IC50 = 240 nM T13127 C6K8WI 11102549 IC50 = 2 nM T13127 CRL01V 11111808 IC50 = 280 nM T13127 CI5OM9 11111827 IC50 = 41 nM T13127 CUPK79 11112773 IC50 = 13 nM T13127 CEPR16 11112815 IC50 = 16200 nM T13127 CK5JA1 11121668 IC50 > 100000 nM T13127 CN3R4Q 11122479 IC50 > 10000 nM T13127 C7P2ZU 11133383 IC50 > 10000 nM T13127 CDZ69K 11133952 IC50 > 10000 nM T13127 CR2E0J 11134506 EC50 = 6 nM T13127 C0VBZ4 11144668 EC50 = 3 nM T13127 CLU8C6 11145028 IC50 = 2.1 nM T13127 CV29TI 11156943 IC50 = 7.2 nM T13127 CH7VS0 11166764 IC50 = 5011.87 nM T13127 CW8GM5 11178452 IC50 = 6300 nM T13127 CAUE56 11178719 EC50 = 9.8 nM T13127 CY52DP 11189976 EC50 = 17.7 nM T13127 CEA1I0 11191318 IC50 = 51 nM T13127 CB5WM8 11202013 IC50 = 220 nM T13127 C3I0AR 11204000 IC50 = 3 nM T13127 CJKQ34 11212886 IC50 = 4073.8 nM T13127 C0J2CG 11224449 IC50 = 1000 nM T13127 C1M5VN 11226024 IC50 = 1400 nM T13127 CG74JV 11237384 IC50 = 1.1 nM T13127 CVM5W4 11237934 IC50 = 2630.27 nM T13127 CP4T9O 11247532 EC50 = 7 nM T13127 CL4JM1 11248965 IC50 = 60 nM T13127 C02PHB 11261604 IC50 = 57000 nM T13127 CT4E5N 11261954 IC50 = 91000 nM T13127 C8Z7LG 11271575 EC50 > 100 nM T13127 C1ECW0 11282348 IC50 = 380 nM T13127 CQ03ZS 11284773 IC50 = 10 nM T13127 CHC58N 11294760 IC50 = 56 nM T13127 CN83IT 11295368 IC50 = 780 nM T13127 C30PBV 11296263 IC50 = 8 nM T13127 CWA42Y 11305084 EC50 = 0.14 nM T13127 CX5F2A 11327727 IC50 = 40738.03 nM T13127 C3AI7K 11327980 EC50 > 100 nM T13127 CT6X5W 11329222 IC50 = 41 nM T13127 CJ2PQ0 11329445 EC50 > 100 nM T13127 C10NUC 11329760 IC50 = 3.4 nM T13127 C2SV7A 11330505 IC50 = 1700 nM T13127 CW03NK 11331099 IC50 = 1000 nM T13127 CUQ2E6 11339578 EC50 > 100 nM T13127 CU60XK 11340002 EC50 = 14 nM T13127 C6T2MI 11352596 EC50 > 100 nM T13127 C08SAG 11361710 EC50 = 140 nM T13127 CPM69O 11362876 EC50 = 13 nM T13127 CI1PU4 11363291 IC50 = 0.3 nM T13127 CQ4R8W 11364483 IC50 = 0.6 nM T13127 CYZ2U1 11364751 IC50 = 79 nM T13127 CVY4S2 11365621 IC50 = 440 nM T13127 C73JGU 11374441 EC50 = 0.81 nM T13127 CSU60Y 11375079 IC50 = 1122.02 nM T13127 CO4YM6 11375135 EC50 = 9.1 nM T13127 COS74H 11376036 IC50 = 5.9 nM T13127 CM41BQ 11376536 IC50 = 321000 nM T13127 C5N6TS 11376932 IC50 = 2200 nM T13127 C9OFN0 11377186 IC50 = 0.4 nM T13127 CC4U0Q 11377266 Ki = 1 nM T13127 CO38NE 11396942 EC50 = 3.3 nM T13127 CQ51LH 11398883 IC50 = 22 nM T13127 C53TQY 11410704 IC50 = 42000 nM T13127 CW1NC3 11419954 EC50 > 100 nM T13127 CB0X7N 11419991 EC50 = 150 nM T13127 CT3GL4 11421054 IC50 = 41 nM T13127 C2PUV0 11430037 EC50 > 100 nM T13127 C2U8AF 11430910 EC50 = 154 nM T13127 C2AZ6M 11430983 EC50 = 15 nM T13127 CZH2W8 11431774 EC50 = 5.1 nM T13127 C7DPE9 11442467 EC50 = 36 nM T13127 CLD17Y 11453686 EC50 = 1 nM T13127 CT5B1R 11454168 EC50 = 130 nM T13127 CT0D2Y 11454792 IC50 = 640 nM T13127 CY8Z6M 11454903 IC50 = 3100 nM T13127 CX0B6H 11456088 IC50 = 6000 nM T13127 CW9DK0 11489353 IC50 = 5 nM T13127 CFYV13 11497803 IC50 = 3000 nM T13127 CP2Y1I 11501268 IC50 > 100000 nM T13127 C7DI5W 11519236 IC50 = 28.5 nM T13127 C6UP1B 11526961 IC50 = 1260 nM T13127 C93QKT 11530057 IC50 > 100000 nM T13127 C9OK1B 11547367 IC50 = 7 nM T13127 C0L9BX 11563200 IC50 = 5500 nM T13127 C50MXC 11569637 IC50 = 1000 nM T13127 C1M0JF 11577483 IC50 = 100 nM T13127 CI3UM9 11577773 IC50 = 10200 nM T13127 C39WPZ 11584551 IC50 = 4300 nM T13127 CCEJ24 11591983 IC50 = 2500 nM T13127 CE03FH 11603180 IC50 > 100000 nM T13127 C1H7IU 11606166 IC50 = 2200 nM T13127 CSF23B 11613911 IC50 > 100000 nM T13127 C3ZXM2 11648999 IC50 = 12.1 nM T13127 CY48MZ 11653900 IC50 = 380 nM T13127 CDIX93 11663899 IC50 = 10500 nM T13127 CJQE01 11671111 IC50 = 4300 nM T13127 C37GDU 11678115 IC50 = 4300 nM T13127 CWQ6H5 11685143 IC50 = 11400 nM T13127 CZBR68 11692944 IC50 = 50 nM T13127 CF4CB6 11705038 IC50 = 0.1 nM T13127 CRZ26B 11710728 IC50 > 100000 nM T13127 C6GYV7 11713906 IC50 = 10300 nM T13127 CF67YA 11726346 IC50 = 9000 nM T13127 CUT1Q0 11728765 IC50 = 2000 nM T13127 CE8HU6 11730182 IC50 = 0.19 nM T13127 C9FBX3 11730503 Ki = 25 nM T13127 CPI13J 11731127 IC50 = 65 nM T13127 CB8N9K 11732098 IC50 = 54 nM T13127 C30TBM 11732162 IC50 = 6800 nM T13127 C6B5AS 11732951 IC50 = 11 nM T13127 CP0YN4 11733318 IC50 = 2140 nM T13127 CF8V0P 11740910 IC50 = 500 nM T13127 CS0P7Z 11753496 IC50 = 160 nM T13127 C64SLQ 11753729 IC50 = 0.32 nM T13127 CQ89UF 11754736 IC50 = 453 nM T13127 C78XPD 11754966 IC50 = 4 nM T13127 CCR1Q5 11755047 IC50 = 570 nM T13127 CHD5A8 11757605 IC50 = 12 nM T13127 C0QT1V 11758430 IC50 = 3800 nM T13127 C1Q8PB 11775366 IC50 = 83176.38 nM T13127 C50NWF 11779696 IC50 = 114 nM T13127 C98XJB 11794292 IC50 = 2800 nM T13127 C9BVU4 11794831 IC50 = 1300 nM T13127 C3SF5M 11796206 IC50 = 200 nM T13127 CD5J4U 11796226 IC50 = 50000 nM T13127 CGP5B4 11796363 IC50 = 80 nM T13127 C8W5XM 11797015 IC50 = 2100 nM T13127 CIT15Q 11797067 IC50 = 4800 nM T13127 CGL25V 11797774 IC50 = 2200 nM T13127 CRB23F 11797967 IC50 = 660 nM T13127 C4OTU6 11798013 IC50 = 1400 nM T13127 CCT82D 11798100 IC50 = 45900 nM T13127 CI46BZ 11798331 IC50 = 580 nM T13127 CZD80O 11798452 IC50 = 10200 nM T13127 CFUC16 11798753 IC50 = 570 nM T13127 C9OBH7 11798777 IC50 = 420 nM T13127 C8ZH3B 11799775 IC50 = 2500 nM T13127 CL2E0S 11799852 IC50 = 920 nM T13127 CA9D2Q 11799888 IC50 = 2500 nM T13127 CZO89U 11800008 IC50 = 6.6 nM T13127 CW3ID0 11800388 IC50 = 50 nM T13127 CI84UQ 11801799 IC50 = 104 nM T13127 CEJ7Z9 11801824 IC50 = 1.8 nM T13127 CJ4TY7 11802020 IC50 = 4300 nM T13127 C0OEA3 11802563 IC50 = 7.9 nM T13127 C7OUJ3 11802564 IC50 = 5.2 nM T13127 CP2U8Z 11812514 IC50 = 0.41 nM T13127 CA4I7V 11824866 IC50 = 370 nM T13127 C5Q2MT 11827520 IC50 = 19 nM T13127 C9YX5M 11827685 IC50 = 69 nM T13127 C70PSM 11974097 IC50 = 310 nM T13127 C9R0FU 12017392 IC50 = 1 nM T13127 CDV4L6 12050403 IC50 = 34 nM T13127 CYV21D 12050404 IC50 = 140 nM T13127 CSN5R4 13059715 IC50 = 2300 nM T13127 CNF98E 13137195 IC50 = 190000 nM T13127 CZC9N7 13661020 IC50 = 79000 nM T13127 CGKE51 14554124 IC50 = 9800 nM T13127 CZ4L9C 14554137 IC50 = 6800 nM T13127 CF7P1W 14885632 IC50 = 56000 nM T13127 CY19RN 15341449 IC50 = 10500 nM T13127 CX79KZ 15390963 IC50 = 495 nM T13127 CGJ85P 15390964 IC50 = 7300 nM T13127 CVGI67 15390974 IC50 = 21 nM T13127 CD6C0M 15410947 IC50 = 950000 nM T13127 C3RQP6 15484952 IC50 = 180 nM T13127 CBA41W 15524013 IC50 > 10000 nM T13127 CL1FK2 15547643 IC50 = 0.56 nM T13127 CPY1L9 15834370 IC50 = 57600 nM T13127 CUY1O9 15839765 IC50 = 470 nM T13127 C29JVP 15839766 IC50 = 2000 nM T13127 CX5L2P 15872083 IC50 = 15 nM T13127 CL4AU7 15949567 IC50 = 0.08 nM T13127 CP0HG4 15967429 IC50 = 3.5 nM T13127 CH68IY 16086144 IC50 = 730 nM T13127 C04LDO 16086145 IC50 = 25 nM T13127 C5JT6Z 16086147 IC50 = 180 nM T13127 CLY6H0 16086150 IC50 = 3700 nM T13127 C5BQ1L 16086151 IC50 = 370 nM T13127 CMPA59 16086153 IC50 = 78 nM T13127 C3S2AI 16086154 IC50 = 390 nM T13127 CY6SC7 16086171 IC50 = 50 nM T13127 CM0HW2 16086173 IC50 = 54 nM T13127 CA8D7C 16086174 IC50 = 114 nM T13127 C4AZ7O 16086175 IC50 = 30 nM T13127 CX59MT 16086178 IC50 = 510 nM T13127 CACQ57 16086179 IC50 = 54 nM T13127 CKEX74 16086181 IC50 = 72 nM T13127 C5CIE8 16086182 IC50 = 370 nM T13127 CFP92T 16086183 IC50 = 230 nM T13127 C8J7KO 16726090 IC50 = 0.01 nM T13127 C3YG0I 16736393 IC50 = 16 nM T13127 CZK80J 16736394 IC50 = 5000 nM T13127 CN80GW 16736585 IC50 = 13 nM T13127 C4BO1G 16760428 IC50 = 2610 nM T13127 CNV1A5 17757984 IC50 = 7.8 nM T13127 CS86PH 17757985 IC50 = 6.5 nM T13127 C9TP2B 17757994 IC50 = 105 nM T13127 CI4Q0K 17758003 IC50 = 10 nM T13127 CS1O4M 17758208 IC50 = 16 nM T13127 CO5J6M 17758316 IC50 = 1.7 nM T13127 C20XEH 17758320 IC50 = 3.2 nM T13127 CF0LQ7 17758323 IC50 = 5.5 nM T13127 CQI9W0 17758430 IC50 = 25 nM T13127 CQY5C7 17759018 IC50 = 7.5 nM T13127 C32TOW 17759286 IC50 = 0.6 nM T13127 CM06OU 17759518 IC50 = 4.8 nM T13127 CS1Y0X 17759638 IC50 = 2.6 nM T13127 CGEY26 17759748 IC50 = 7 nM T13127 C6U9DY 17900419 IC50 = 16 nM T13127 CI0X3S 17900438 IC50 = 65 nM T13127 CX28RA 17900448 IC50 = 115 nM T13127 CBZQ34 17900480 IC50 = 150 nM T13127 C2ZV3N 17900489 IC50 = 720 nM T13127 CD3SH1 17900490 IC50 = 88 nM T13127 CX8ZG7 17900495 IC50 = 30 nM T13127 CCQU32 17900499 IC50 = 32 nM T13127 CRX15A 17900521 IC50 = 100 nM T13127 C80JFP 17965976 IC50 = 1.4 nM T13127 CITW75 18177056 IC50 = 3 nM T13127 CN7Q2W 18177084 IC50 = 2.8 nM T13127 CQ68EN 18177125 IC50 = 2.5 nM T13127 C2RX1W 18391309 Ki = 140 nM T13127 CJ2T8C 18391310 Ki = 738 nM T13127 CO24YD 18431465 IC50 = 6 nM T13127 CSFH45 18433542 IC50 = 10 nM T13127 C2SEG5 18433574 IC50 = 2.5 nM T13127 CW27VZ 18475821 IC50 = 15 nM T13127 C8PW9F 18475830 IC50 = 5.7 nM T13127 C7BIR8 18475867 IC50 = 2.5 nM T13127 CP9IG3 18536049 IC50 = 38 nM T13127 C7C9JU 18536050 IC50 = 1.2 nM T13127 CWDQ78 18536130 IC50 = 0.66 nM T13127 CD4F6M 18536154 IC50 = 20 nM T13127 C7X1OV 18536181 IC50 = 0.31 nM T13127 C0YLC9 18670809 IC50 = 500 nM T13127 CK2P3O 18715188 IC50 = 2100 nM T13127 CQ4GB7 18715194 IC50 = 2000 nM T13127 C4BG7H 18715214 IC50 = 2100 nM T13127 C7JXY0 18715403 IC50 = 724000 nM T13127 C85LBY 20585594 IC50 = 170 nM T13127 CD3EU4 20585595 IC50 = 6.8 nM T13127 C8HQ7K 20585599 IC50 = 645 nM T13127 CL4MG1 20585601 IC50 = 0.26 nM T13127 CS5F1D 20585631 IC50 = 0.86 nM T13127 C2JY1H 20585632 IC50 = 1.4 nM T13127 CAWR19 20585634 IC50 = 0.1 nM T13127 CWH59K 20585639 IC50 = 19 nM T13127 C1FPD5 20622765 IC50 = 0.21 nM T13127 CX4LN5 20622881 IC50 = 0.58 nM T13127 C1FXV8 20622885 IC50 = 0.92 nM T13127 CKG3M0 20622887 IC50 = 0.81 nM T13127 CP4U5B 20622889 IC50 = 12 nM T13127 C2QI7V 20622895 IC50 = 26 nM T13127 C0ZW4K 20638589 IC50 = 1 nM T13127 CD6S5T 20659966 IC50 = 2300 nM T13127 CQ8CL9 20691443 IC50 = 86 nM T13127 CX5SM9 21082040 IC50 = 6 nM T13127 CNT0Q4 21082041 IC50 = 26 nM T13127 C2HW5C 21082080 IC50 = 1.3 nM T13127 C4PWD1 21197625 IC50 = 5000 nM T13127 CU1NR6 21197628 IC50 > 10000 nM T13127 C35GYP 21680425 IC50 > 40000 nM T13127 C9J5CA 21696948 IC50 = 38 nM T13127 C0OD7R 21696958 IC50 = 110 nM T13127 CODT84 21696968 IC50 = 180 nM T13127 C0SL1P 21696982 IC50 = 100 nM T13127 COS78Y 21696999 IC50 = 38 nM T13127 C4F1XV 21697006 IC50 = 17 nM T13127 C72TUJ 21697011 IC50 = 14 nM T13127 CT52HZ 21697013 IC50 = 41 nM T13127 CIZ28U 21697015 IC50 = 45 nM T13127 C7CJ1S 21697020 IC50 = 230 nM T13127 CH5G2U 21697037 IC50 = 27 nM T13127 C05JIL 21697038 IC50 = 5400 nM T13127 CC27MY 21697040 IC50 = 290 nM T13127 CX7K6O 21697048 IC50 = 1500 nM T13127 C2Q3GM 21697057 IC50 = 8 nM T13127 CLP87G 21697066 IC50 = 390 nM T13127 CAZ1Y8 21697070 IC50 = 38 nM T13127 C6MUK9 21697098 IC50 = 28 nM T13127 CI43WK 21697104 IC50 = 130 nM T13127 C3RFE7 21697108 IC50 = 38 nM T13127 CF75LI 21697118 IC50 = 40 nM T13127 C0L4KV 21697122 IC50 = 150 nM T13127 C1FKS0 21697124 IC50 = 27 nM T13127 C69SUH 21697133 IC50 = 340 nM T13127 C1TD9Y 22082992 IC50 = 16 nM T13127 C0KRU8 22082993 IC50 = 1.8 nM T13127 C9WP8T 22082994 IC50 = 3.3 nM T13127 C1QZS6 22082995 IC50 = 18 nM T13127 CU5J9R 22083000 IC50 = 50 nM T13127 CD0ZO5 22404047 IC50 = 880 nM T13127 C1TS5R 22466803 IC50 = 0.2 nM T13127 C4XBJ1 22466804 IC50 = 0.21 nM T13127 C2CMD3 22466823 IC50 = 0.7 nM T13127 COI40N 22466825 IC50 = 1.1 nM T13127 C17IKZ 22466836 IC50 = 0.9 nM T13127 CW49TR 22466839 IC50 = 2.1 nM T13127 C0GN4Z 22466842 IC50 = 7.7 nM T13127 C9I4PY 22466854 IC50 = 1.2 nM T13127 CWD2A4 22466855 IC50 = 0.5 nM T13127 C2MN0S 22466859 IC50 = 1.7 nM T13127 CNYM47 22466875 IC50 = 0.16 nM T13127 CW3FH0 22466880 IC50 = 0.35 nM T13127 CM8K2E 22466884 IC50 = 0.73 nM T13127 CX7E4O 22466886 IC50 = 0.37 nM T13127 CZ5X2G 22466888 IC50 = 0.72 nM T13127 CB1AD5 22466891 IC50 = 0.24 nM T13127 C8A4NF 22466894 IC50 = 1.3 nM T13127 C3Y2WH 22466895 IC50 = 0.09 nM T13127 C70PSA 22466899 IC50 = 0.75 nM T13127 CI6B0M 22621920 IC50 = 1140 nM T13127 C8BID3 22625935 IC50 = 18 nM T13127 C6ZA0X 22744657 IC50 = 108 nM T13127 CWX91B 22884086 IC50 = 160 nM T13127 COP68C 22914796 IC50 = 22300 nM T13127 CR9BC0 22921993 IC50 > 11000 nM T13127 CH3PO5 22966419 IC50 = 4.9 nM T13127 CJ81SY 23289845 IC50 = 1120 nM T13127 CHL2X5 23289847 IC50 = 61 nM T13127 CT54IB 23289866 IC50 = 140 nM T13127 C0M2NX 23289901 IC50 = 1100 nM T13127 CMZN30 23289903 IC50 = 32 nM T13127 CY84AM 23388879 IC50 = 1.5 nM T13127 C9B1YI 23388975 IC50 = 5 nM T13127 CV4XB8 23388978 IC50 = 3 nM T13127 CBV19H 23425708 IC50 = 21510 nM T13127 C0T8EZ 23427323 IC50 > 30000 nM T13127 CVO8M3 23575252 IC50 = 96.5 nM T13127 CHO7L4 23575254 IC50 = 61 nM T13127 C03VZX 23575255 IC50 = 53.2 nM T13127 C5T7BA 23575256 IC50 = 89.3 nM T13127 CC92BR 23575257 IC50 = 28.3 nM T13127 C38WGU 23575258 IC50 = 26 nM T13127 CAJH43 23575319 IC50 = 19 nM T13127 C2Q3EH 23575320 IC50 = 75 nM T13127 C1O4UD 23575326 IC50 = 44 nM T13127 C7ZJ1F 23633300 IC50 > 100000 nM T13127 C75XYD 23643216 IC50 = 299 nM T13127 CY32DX 23643650 IC50 = 60000 nM T13127 C9KU7R 23646369 IC50 = 20400 nM T13127 CS6Z3R 23646370 IC50 = 70500 nM T13127 CUJ0D3 23646577 IC50 = 1.6 nM T13127 C2YL0F 23647730 IC50 = 2.5 nM T13127 C26PFW 23647731 IC50 = 0.71 nM T13127 CX03NL 23647732 IC50 = 560 nM T13127 C1Y6NX 23647733 IC50 = 280 nM T13127 CHZ2P0 23647734 IC50 = 240 nM T13127 CTR64K 23647735 IC50 = 310 nM T13127 CMV6E8 23708717 EC50 > 1 nM T13127 CY2QO1 23708724 EC50 = 0.9 nM T13127 C1D8YT 24180547 IC50 = 17.3 nM T13127 CFEA98 24809846 IC50 = 5.5 nM T13127 C3XU6B 25053256 IC50 = 420 nM T13127 C7I3VM 25053455 IC50 = 1000 nM T13127 CZ46WT 25053523 IC50 = 450 nM T13127 CGK60P 25053583 IC50 = 650 nM T13127 CBPE64 25053639 IC50 = 380 nM T13127 CZ7XH0 25141073 IC50 = 1.5 nM T13127 CU86ET 25256804 IC50 = 1.1 nM T13127 CEJ21Y 44266892 IC50 = 20 nM T13127 CBUI64 44266894 IC50 = 12 nM T13127 CO6N7A 44266896 IC50 = 8.4 nM T13127 CY5SM1 44266936 IC50 = 560 nM T13127 CK0ZD4 44266942 IC50 = 9.9 nM T13127 CPAM05 44266949 IC50 > 1000 nM T13127 CZWQ45 44266950 IC50 = 6 nM T13127 C76DKF 44266955 IC50 = 19 nM T13127 CNQ62C 44266958 IC50 = 41000 nM T13127 C90IAD 44266964 IC50 = 1.2 nM T13127 CYSK72 44266966 IC50 = 6.6 nM T13127 C7V9YZ 44266972 IC50 = 8.8 nM T13127 C7WB0M 44266976 EC50 = 0.3 nM T13127 C5AEO0 44266979 IC50 = 3 nM T13127 C53HZA 44266980 IC50 = 2.4 nM T13127 C0ZVB8 44266982 EC50 = 1.2 nM T13127 CF81VP 44266988 EC50 = 10 nM T13127 CHU17O 44266992 EC50 = 1.8 nM T13127 C7XU9R 44266994 EC50 = 1.5 nM T13127 CZR32K 44266996 EC50 = 0.1 nM T13127 CBF4Q9 44266998 IC50 = 6.3 nM T13127 C3WZ5F 44267003 EC50 = 0.78 nM T13127 CIDM13 44267017 EC50 = 10 nM T13127 CBP4L0 44267022 IC50 = 4.9 nM T13127 C74LVI 44274781 EC50 = 7.9 nM T13127 C34TGF 44274782 IC50 = 0.68 nM T13127 C4XQY2 44274783 EC50 < 1 nM T13127 C2PNA5 44274804 EC50 = 9.8 nM T13127 C2U0NZ 44274806 IC50 = 3.3 nM T13127 CA9MJ4 44274825 IC50 = 33 nM T13127 C38NIZ 44276567 IC50 = 900 nM T13127 C5I8SU 44276702 IC50 = 68 nM T13127 CK41CL 44276714 IC50 = 24 nM T13127 C8H9ER 44277448 IC50 = 59 nM T13127 CLZ60X 44277454 IC50 = 0.5 nM T13127 COB19E 44277466 IC50 = 15 nM T13127 CLI62D 44277527 IC50 = 3.5 nM T13127 CVEM18 44277528 IC50 = 3.1 nM T13127 C4D6QO 44277534 IC50 = 0.5 nM T13127 CFRL98 44277536 IC50 = 20 nM T13127 C7C0SX 44277543 IC50 = 35 nM T13127 CJI3Q4 44279741 IC50 = 255 nM T13127 CR9P0Z 44279816 IC50 = 4000 nM T13127 CHGQ78 44279912 IC50 = 670 nM T13127 CW3Q2R 44279932 IC50 = 1230 nM T13127 CA2F7Q 44279976 IC50 = 48 nM T13127 CLS53M 44280014 IC50 = 5770 nM T13127 C2Z0ED 44280183 IC50 >> 10000 nM T13127 C7GO4Y 44282173 IC50 = 10000 nM T13127 CUTC61 44282252 IC50 = 5000 nM T13127 CM6PG1 44282288 IC50 = 190 nM T13127 C0WPI4 44282393 IC50 = 900 nM T13127 CRU05G 44282588 IC50 > 10000 nM T13127 CI83JG 44282596 IC50 = 1000 nM T13127 C4ET5R 44285512 IC50 = 3.5 nM T13127 C1OXU5 44286155 IC50 = 1.7 nM T13127 CU6PI8 44286156 IC50 = 22 nM T13127 C34UPR 44286166 IC50 = 48 nM T13127 CLT5M7 44286182 IC50 = 6 nM T13127 CUR1S4 44286305 IC50 = 4 nM T13127 CLRV12 44286360 IC50 = 1.6 nM T13127 CRKC91 44287977 IC50 = 3400 nM T13127 C3Z1BP 44294472 IC50 = 10100 nM T13127 C5TQ3S 44294487 IC50 = 453 nM T13127 CXSH90 44294608 IC50 = 17 nM T13127 COC3R7 44294615 IC50 = 2220 nM T13127 CM9VL4 44294641 IC50 = 290 nM T13127 C28PQY 44294653 IC50 = 102 nM T13127 CNO8T5 44294666 IC50 = 1400 nM T13127 C2XTW0 44294675 IC50 = 6600 nM T13127 C0ZH6D 44294959 IC50 = 950 nM T13127 CBD01X 44296738 Ki = 25500 nM T13127 C8F0XJ 44296739 Ki = 32000 nM T13127 C7UPK1 44296753 IC50 = 6.6 nM T13127 C0CI8N 44296765 Ki = 40000 nM T13127 CE52FL 44296772 IC50 = 3.8 nM T13127 C2YN8J 44296782 Ki = 50000 nM T13127 C0FWV4 44296784 IC50 = 8 nM T13127 C4XVQ5 44296801 Ki = 420 nM T13127 CCX94L 44296840 Ki = 420 nM T13127 CNT13I 44296869 Ki = 250 nM T13127 C7MWN2 44296940 IC50 = 2.7 nM T13127 C9OT0J 44296947 IC50 = 7 nM T13127 CC6R0J 44297001 IC50 = 2.3 nM T13127 C94AVI 44297038 IC50 = 1.2 nM T13127 C51STW 44297041 IC50 = 2.1 nM T13127 CB17VJ 44298237 IC50 = 200 nM T13127 CC5LT6 44298380 EC50 = 0.18 nM T13127 CP6Z9A 44298623 IC50 = 1000 nM T13127 CXQD94 44298864 IC50 = 200 nM T13127 CHG2P4 44298887 IC50 > 360000 nM T13127 CK93WE 44298915 IC50 > 360000 nM T13127 C31KRW 44298943 IC50 = 166000 nM T13127 C71XHO 44298944 IC50 = 63000 nM T13127 CY5ZQ7 44298951 IC50 > 360000 nM T13127 CA2YH8 44298963 IC50 = 157000 nM T13127 CS7GU9 44298991 IC50 = 137000 nM T13127 C85PNQ 44299002 IC50 > 360000 nM T13127 C15XEF 44299016 IC50 > 360000 nM T13127 CKZ8V7 44299018 IC50 = 29000 nM T13127 CGQ59J 44302675 IC50 = 80000 nM T13127 CN7CX2 44302690 IC50 = 870 nM T13127 C86SOA 44302691 IC50 = 55 nM T13127 CF8D6O 44302699 IC50 = 183 nM T13127 C1E3ZG 44302700 IC50 = 260 nM T13127 C4I7TY 44302717 IC50 = 1075 nM T13127 CZX61D 44302764 IC50 = 300 nM T13127 C0DNT3 44302842 IC50 = 12000 nM T13127 C38JPF 44302867 IC50 = 1750 nM T13127 C8W2GF 44302875 IC50 = 255 nM T13127 CY10HD 44302886 IC50 = 58 nM T13127 C1CRS4 44302887 IC50 = 355 nM T13127 CKEZ67 44302927 IC50 = 23 nM T13127 CAX98M 44302928 IC50 = 27 nM T13127 CH1XF2 44302953 IC50 = 12 nM T13127 CL8I1C 44303006 IC50 = 14 nM T13127 C6P0ZJ 44303744 IC50 = 0.85 nM T13127 C8CJ0O 44304028 IC50 = 6.8 nM T13127 C8F9BE 44304133 IC50 = 6.1 nM T13127 C14JQT 44304150 IC50 = 3.17 nM T13127 C8E9GQ 44305558 IC50 = 460000 nM T13127 CCJY27 44306966 IC50 = 20000 nM T13127 C6YX7J 44306967 IC50 = 1800 nM T13127 CY3W1U 44306968 IC50 = 10000 nM T13127 CHQ8S5 44306989 IC50 = 33 nM T13127 CQ7FC6 44306990 IC50 = 150 nM T13127 CVP9R0 44307001 IC50 > 360000 nM T13127 C0G9LA 44307003 IC50 > 360000 nM T13127 C50MIK 44307004 IC50 = 1200 nM T13127 CTOQ60 44307005 IC50 = 900 nM T13127 CU1YH7 44307053 IC50 = 4500 nM T13127 CN5Y2B 44307395 IC50 = 4400 nM T13127 CTY27X 44315100 IC50 = 1.8 nM T13127 CIP1H8 44315132 IC50 = 1.4 nM T13127 C8K0TX 44315147 IC50 = 85 nM T13127 CEM8B5 44315148 IC50 = 0.46 nM T13127 CGKU37 44315154 IC50 = 0.57 nM T13127 C4F6AJ 44315320 IC50 = 0.75 nM T13127 CI4OE7 44315339 IC50 = 0.37 nM T13127 CH4B1V 44315359 IC50 = 120 nM T13127 CS8NG0 44315440 IC50 = 3900 nM T13127 C0HQ4D 44315459 IC50 = 14 nM T13127 COJS30 44315505 IC50 = 4.4 nM T13127 CRLO35 44315546 IC50 = 90 nM T13127 CI7PH8 44315549 IC50 = 45 nM T13127 CBR1W4 44315551 IC50 = 5300 nM T13127 CE65ON 44315563 IC50 = 270 nM T13127 C2H7RY 44315577 IC50 = 37 nM T13127 C67ZKP 44315601 IC50 = 0.6 nM T13127 C9ACR7 44315661 IC50 = 2.8 nM T13127 C7E3LC 44315772 IC50 = 0.92 nM T13127 CBL41F 44315773 IC50 = 770 nM T13127 CQ2G4J 44315787 IC50 = 1 nM T13127 CT7NW1 44315827 IC50 = 160 nM T13127 CW94FB 44315828 IC50 = 1100 nM T13127 CASW94 44315829 IC50 = 8200 nM T13127 CIKR68 44317074 IC50 = 23 nM T13127 C7ZP9T 44317169 IC50 = 1.4 nM T13127 C5FQH4 44317319 EC50 = 1 nM T13127 C3RN4G 44317321 IC50 = 170 nM T13127 CZ5A4P 44317414 IC50 = 0.06 nM T13127 C0VXH7 44318498 IC50 = 5000 nM T13127 CILZ87 44318666 IC50 = 2100 nM T13127 CHS90P 44318863 IC50 = 20000 nM T13127 C68QBX 44318864 IC50 = 840 nM T13127 C4BU8T 44318866 IC50 = 3400 nM T13127 CVOX30 44318867 IC50 = 1000 nM T13127 C46OUP 44318880 IC50 = 140 nM T13127 C2O6SK 44318894 IC50 = 79 nM T13127 C6D4ZC 44320292 IC50 = 14000 nM T13127 C5G9AK 44320314 IC50 = 100000 nM T13127 C7J2IO 44320337 IC50 = 100000 nM T13127 C7TKZ8 44320418 IC50 = 18000 nM T13127 CKZI07 44320678 IC50 > 1000000 nM T13127 CQS21A 44320873 IC50 > 1000000 nM T13127 C9KU2Q 44323670 IC50 = 2000 nM T13127 C0OV7B 44323677 IC50 > 100000 nM T13127 C7UK6V 44323743 IC50 = 5 nM T13127 CG58AC 44323747 IC50 > 100000 nM T13127 C05YVE 44323748 IC50 = 50 nM T13127 C4W6GV 44323761 IC50 > 100000 nM T13127 C3SZ7N 44323961 IC50 = 100 nM T13127 CMG5D0 44323963 IC50 > 100000 nM T13127 CK0PY3 44323964 IC50 = 290 nM T13127 CE4G9W 44326397 IC50 = 105 nM T13127 CRU0Z4 44326554 IC50 = 20400 nM T13127 CZDQ40 44326555 IC50 = 6600 nM T13127 CRU53F 44326556 IC50 = 1860 nM T13127 C8L1CS 44326557 IC50 = 32 nM T13127 CJN3R7 44326562 IC50 = 16 nM T13127 C02LEV 44326590 IC50 = 7 nM T13127 C7S0VO 44326598 IC50 = 18 nM T13127 CT62RE 44326618 IC50 = 16 nM T13127 CBD31T 44326619 IC50 = 3300 nM T13127 CCX6W9 44326642 IC50 = 80 nM T13127 CDC6H9 44326643 IC50 = 1200 nM T13127 CX1A6E 44326679 IC50 = 230 nM T13127 CQ2B7X 44326680 IC50 = 940 nM T13127 CMWY28 44326695 IC50 = 240 nM T13127 C3B5XC 44326720 IC50 = 9 nM T13127 C4R7ZG 44326726 IC50 = 315 nM T13127 CRK84G 44326729 IC50 = 170 nM T13127 CUNV12 44326835 IC50 = 9700 nM T13127 COR6H3 44326873 IC50 = 1000 nM T13127 CG3QU9 44326874 IC50 = 1900 nM T13127 CAG1O4 44326875 IC50 = 33 nM T13127 CGQ30P 44331329 IC50 = 1350 nM T13127 C3VB9L 44331330 IC50 = 470 nM T13127 CXUC31 44331375 IC50 = 5000 nM T13127 CUSE79 44331378 IC50 = 2300 nM T13127 C6P9UY 44331590 IC50 = 3050 nM T13127 C2O9AR 44331720 IC50 > 12000 nM T13127 CL0TE5 44331801 IC50 = 1200 nM T13127 C4XBP1 44331807 IC50 > 10000 nM T13127 C4SQR2 44331808 IC50 = 4800 nM T13127 CY2RM4 44331820 IC50 = 3600 nM T13127 C6L7WD 44331846 IC50 > 10000 nM T13127 CYU9R7 44331851 IC50 > 10000 nM T13127 C4GH6Y 44331867 IC50 = 4700 nM T13127 CP6J7E 44331906 IC50 = 8500 nM T13127 CY8U0A 44331909 IC50 = 8800 nM T13127 CT4CI7 44331924 IC50 = 6290 nM T13127 CVX13Y 44331945 IC50 = 4800 nM T13127 C40WON 44331946 IC50 = 5200 nM T13127 C4GD9H 44331952 IC50 > 12000 nM T13127 C48OTC 44331959 IC50 = 1900 nM T13127 C62GWV 44331960 IC50 = 4600 nM T13127 CA0TM4 44332063 IC50 = 13000 nM T13127 C1C4YE 44332070 IC50 = 8400 nM T13127 C7R6FH 44332086 IC50 = 9600 nM T13127 C1O3HS 44332094 IC50 > 12000 nM T13127 C8XB6C 44332095 IC50 = 10600 nM T13127 CZ3A8H 44332114 IC50 = 8200 nM T13127 CKC45E 44332130 IC50 = 11400 nM T13127 C18JUG 44332210 IC50 = 20 nM T13127 CT3R7H 44332263 IC50 = 75 nM T13127 C0L4WQ 44332321 IC50 = 50 nM T13127 C1Z9NA 44332322 IC50 = 0.5 nM T13127 CRG4F8 44332323 IC50 = 60 nM T13127 CT7AZ4 44332326 IC50 = 83 nM T13127 CL2YV3 44332383 IC50 = 185 nM T13127 CUJ9G3 44332403 IC50 = 100 nM T13127 CC2E1Z 44334508 IC50 = 2000 nM T13127 C2Q3GC 44334509 IC50 = 2.1 nM T13127 CCK79N 44336289 IC50 = 5.4 nM T13127 CCS87O 44340658 IC50 = 525 nM T13127 C5WE3U 44340738 IC50 > 10000 nM T13127 C76FXG 44340755 IC50 = 310 nM T13127 C3Y8OK 44340756 IC50 = 230 nM T13127 C5-JAN-01 44340757 IC50 = 14 nM T13127 CHIF54 44340776 IC50 = 37 nM T13127 CSJ53C 44340777 IC50 = 19 nM T13127 CNQ3E5 44340778 IC50 = 6.2 nM T13127 CLX9G7 44340791 IC50 = 0.123 nM T13127 C9WCV0 44340884 IC50 = 29 nM T13127 CT21QH 44340933 IC50 = 230 nM T13127 C3TH9I 44340934 IC50 = 51 nM T13127 C0G8XN 44340935 IC50 = 36 nM T13127 CMXL69 44340936 IC50 = 260 nM T13127 CU24RJ 44340937 IC50 = 230 nM T13127 C3BD9G 44340938 IC50 = 17 nM T13127 CACB20 44340960 IC50 > 10000 nM T13127 CG80UI 44340975 IC50 > 10000 nM T13127 C4Q3NR 44340977 IC50 = 16 nM T13127 CGK1I7 44340978 IC50 = 17 nM T13127 CBP0N6 44340982 IC50 = 160 nM T13127 CZP0C1 44340983 IC50 = 120 nM T13127 CQ73AL 44341007 IC50 = 23 nM T13127 CY9BN1 44341008 IC50 = 86 nM T13127 CEL34B 44341009 IC50 = 70 nM T13127 CN5EV4 44341025 IC50 = 190 nM T13127 C2QSD8 44341660 IC50 = 13 nM T13127 CZ81FE 44341671 IC50 430 nM T13127 C30COY 44341758 IC50 = 2.8 nM T13127 CJB79M 44341773 IC50 = 0.41 nM T13127 C54EXR 44341781 IC50 = 0.12 nM T13127 CJ2VB6 44341788 IC50 = 0.12 nM T13127 C2MNZ5 44341842 IC50 = 4 nM T13127 C0SGE6 44341854 IC50 = 2.8 nM T13127 C31-JAN 44341885 IC50 = 0.15 nM T13127 C3NB1G 44341886 IC50 = 10 nM T13127 C7Q3BF 44341888 IC50 = 74 nM T13127 C8JM1N 44341889 IC50 = 82 nM T13127 C0A7NT 44341933 IC50 = 0.16 nM T13127 C1QF2D 44341960 IC50 = 0.55 nM T13127 C0XEA8 44342060 IC50 = 0.45 nM T13127 CSUK30 44345348 IC50 = 4.4 nM T13127 CXLM82 44345349 IC50 = 28 nM T13127 C7BYE4 44345485 IC50 = 6800 nM T13127 CJ12QM 44345486 IC50 = 20 nM T13127 C3UAB1 44345487 IC50 = 3.4 nM T13127 CCT32K 44346734 IC50 > 100000 nM T13127 C6ZOU8 44346735 IC50 > 100000 nM T13127 CDE8C3 44346895 IC50 > 100000 nM T13127 CJP6C0 44347007 IC50 > 100000 nM T13127 CY6DA7 44348773 IC50 = 0.18 nM T13127 C48IJR 44348932 IC50 = 1 nM T13127 C7N1YP 44349167 IC50 > 0.15 nM T13127 CU6C1L 44349507 IC50 = 0.63 nM T13127 CC80LB 44349537 IC50 = 215 nM T13127 CQAR61 44349693 IC50 = 0.9 nM T13127 CB2Y9E 44349708 IC50 = 1.4 nM T13127 C1D7PV 44349709 IC50 = 0.62 nM T13127 CW5F1L 44349711 IC50 = 2.9 nM T13127 CUQ0T3 44349887 IC50 = 0.61 nM T13127 CFA9V5 44349898 IC50 = 1.1 nM T13127 CI50EZ 44349903 IC50 = 1.3 nM T13127 C3SV8M 44349906 IC50 = 1.6 nM T13127 CJ54FV 44349911 IC50 = 0.55 nM T13127 C9QFW5 44349918 IC50 = 1.3 nM T13127 C02GDH 44349923 IC50 = 0.87 nM T13127 CP9WA5 44349924 IC50 = 1.7 nM T13127 CFL5V1 44349925 IC50 = 0.95 nM T13127 CB0EH3 44349978 IC50 = 10 nM T13127 C1OC4X 44349979 IC50 = 1 nM T13127 CE18FW 44350296 IC50 = 42 nM T13127 CS06LR 44350297 IC50 = 34 nM T13127 C9U1OQ 44350405 IC50 = 2.6 nM T13127 C7IFQ0 44352132 IC50 = 0.49 nM T13127 C19ERO 44352143 EC50 = 1.2 nM T13127 CGX0N1 44352211 EC50 = 11 nM T13127 CJ84GE 44352228 EC50 = 39 nM T13127 CZV91R 44352229 IC50 = 0.42 nM T13127 CNXU54 44352231 IC50 = 9.9 nM T13127 CK3JR1 44352258 IC50 = 0.69 nM T13127 CV03ZL 44352314 IC50 = 1.1 nM T13127 CQ0H6P 44352315 IC50 = 2.7 nM T13127 CRD47I 44352325 IC50 = 5.5 nM T13127 CG6HT2 44352327 EC50 = 17 nM T13127 C79OFM 44352330 IC50 = 6.5 nM T13127 C9T5OF 44352336 EC50 = 10 nM T13127 C5ME4L 44352337 IC50 = 6.3 nM T13127 CU0A8D 44352343 IC50 = 2 nM T13127 CJNY34 44352355 IC50 = 6.1 nM T13127 CFN8G4 44352367 IC50 = 0.42 nM T13127 CZM6E0 44352378 IC50 = 0.51 nM T13127 C4YT1L 44352388 EC50 = 10 nM T13127 CR9DA3 44352390 EC50 = 15 nM T13127 CU3N1R 44352395 IC50 = 0.73 nM T13127 CS84UY 44352396 EC50 = 0.81 nM T13127 C5VL6E 44352409 EC50 = 16 nM T13127 C61DSL 44352416 EC50 = 4.7 nM T13127 C5K4MA 44352423 IC50 = 71 nM T13127 CH50DK 44352429 EC50 = 21 nM T13127 CC1R2H 44352430 IC50 = 1.3 nM T13127 CC1B4K 44352432 EC50 = 4.8 nM T13127 CTC8Q5 44352434 IC50 = 0.036 nM T13127 C6CRZ2 44352446 IC50 = 0.73 nM T13127 CB58TW 44352456 IC50 = 3.9 nM T13127 CF4W2J 44352459 IC50 = 5.3 nM T13127 CH4T5I 44352461 IC50 = 0.81 nM T13127 CWZN84 44352463 EC50 = 24 nM T13127 CSN0P3 44352470 IC50 = 0.75 nM T13127 CZ8R9X 44352471 IC50 = 1.9 nM T13127 CGS09J 44352475 IC50 = 0.85 nM T13127 CSZ4V9 44353707 IC50 = 3200 nM T13127 CMD6A1 44353723 IC50 = 1400 nM T13127 CKJ1R7 44353729 IC50 <= 5000 nM T13127 C7BA8U 44353914 IC50 = 5000 nM T13127 C9RUB5 44353915 IC50 = 2300 nM T13127 CY0XD7 44353928 IC50 = 1832000 nM T13127 CNCU42 44353929 IC50 = 48400 nM T13127 CP86OE 44353931 IC50 = 14900 nM T13127 CT5K2Q 44353932 IC50 = 5300 nM T13127 CS0C7H 44353948 IC50 = 10700 nM T13127 CI6J4P 44353950 IC50 = 1000 nM T13127 CP6S3Z 44353971 IC50 = 32700 nM T13127 CU92NC 44353979 IC50 = 1800 nM T13127 CBMT25 44353997 IC50 = 700 nM T13127 CNM06J 44354002 IC50 = 870 nM T13127 CNRT35 44354012 IC50 = 34000 nM T13127 CIL3G9 44356437 IC50 = 2500 nM T13127 CEKC85 44357811 IC50 = 4 nM T13127 C0ACH2 44358859 IC50 = 6.6 nM T13127 CXA4B8 44359336 IC50 = 1200 nM T13127 C1W3KM 44359339 IC50 = 50000 nM T13127 C6SH2Y 44359345 IC50 = 1200 nM T13127 C4FT3B 44359346 IC50 = 96000 nM T13127 C91LIE 44359351 IC50 > 100000 nM T13127 C20MGJ 44359379 IC50 = 12000 nM T13127 CYV9I4 44359380 IC50 = 38000 nM T13127 CA1FS0 44359391 IC50 > 100000 nM T13127 CY1Q6K 44359406 IC50 > 100000 nM T13127 CY40BM 44359416 IC50 = 40000 nM T13127 C6BY9W 44359426 IC50 = 40 nM T13127 CVS38F 44359434 IC50 = 60000 nM T13127 CY29JN 44359435 IC50 = 3000 nM T13127 C5HK2P 44359440 IC50 > 100000 nM T13127 CF7MA6 44359450 IC50 = 40000 nM T13127 CYS9J6 44359468 IC50 = 21000 nM T13127 C2JZ3T 44359469 IC50 = 31000 nM T13127 CC91FR 44359480 IC50 = 8000 nM T13127 CW3D1R 44359483 IC50 > 100000 nM T13127 C3I8FD 44359513 IC50 = 48000 nM T13127 CGI42H 44359527 IC50 = 40000 nM T13127 C38LBG 44359595 IC50 = 24000 nM T13127 CRH16I 44359602 IC50 = 29000 nM T13127 C40OEX 44359604 IC50 > 100000 nM T13127 CMKE51 44359605 IC50 > 100000 nM T13127 C48GBR 44359635 IC50 = 40000 nM T13127 CW4MC0 44359642 IC50 > 100000 nM T13127 C9VX2Q 44359694 IC50 > 100000 nM T13127 C6IEA9 44359702 IC50 = 56000 nM T13127 C5NHR3 44359713 IC50 = 15000 nM T13127 C78BFK 44359721 IC50 > 100000 nM T13127 C6SBU4 44359727 IC50 = 6800 nM T13127 C5WT4V 44359728 IC50 = 26000 nM T13127 CCOZ12 44366553 IC50 = 34 nM T13127 CQN2U7 44366894 IC50 = 20 nM T13127 C4UPF0 44367161 IC50 = 21000 nM T13127 CP1A5S 44367183 IC50 = 250000 nM T13127 C5GC1I 44367240 IC50 = 16000 nM T13127 CCV36W 44367241 IC50 = 5000 nM T13127 CKW56E 44367281 IC50 = 33000 nM T13127 CW9KX0 44367282 IC50 = 11000 nM T13127 C9Z7BG 44370346 IC50 = 100 nM T13127 C5P1VY 44370348 IC50 = 116 nM T13127 C5R0LZ 44370360 IC50 = 32 nM T13127 CN9Z1Y 44370373 IC50 = 320 nM T13127 CML9U5 44370478 IC50 = 29 nM T13127 CH7ML1 44370508 IC50 = 230 nM T13127 CM2OQ8 44370517 IC50 = 43 nM T13127 CNV4M9 44370539 IC50 = 82 nM T13127 C2F5CX 44370577 IC50 = 62 nM T13127 C5CP3B 44370587 IC50 = 170 nM T13127 CRF7S1 44370619 IC50 = 150 nM T13127 CTSD98 44370620 IC50 = 105 nM T13127 CI5T9R 44370628 IC50 = 199 nM T13127 CDM7W4 44370674 IC50 = 18 nM T13127 CPNZ60 44370676 IC50 = 6 nM T13127 CZRX47 44370691 IC50 = 15800 nM T13127 CYEX16 44370708 IC50 = 260 nM T13127 C1E5MJ 44370714 IC50 = 38 nM T13127 CWH8P7 44370716 IC50 = 84 nM T13127 CIC7Z8 44370717 IC50 = 74 nM T13127 CHUE23 44370720 IC50 = 35 nM T13127 CN9FH3 44370721 IC50 = 240 nM T13127 CCGZ61 44370726 IC50 = 58 nM T13127 C5Q4VK 44370762 IC50 = 15 nM T13127 CF1C2P 44370763 IC50 = 124 nM T13127 C4ND7W 44370811 IC50 = 43 nM T13127 CR9AP1 44370828 IC50 = 6 nM T13127 C4ZHC9 44370830 IC50 < 110 nM T13127 CKD8O5 44370963 IC50 = 8.2 nM T13127 C3I8LQ 44370968 IC50 = 86 nM T13127 C3BG2C 44370976 IC50 = 30 nM T13127 CVT59F 44371659 EC50 = 96 nM T13127 CG7E2K 44372665 IC50 < 1 nM T13127 C62QCE 44372679 IC50 = 24 nM T13127 CNEK75 44372893 IC50 < 1 nM T13127 CE5AQ0 44375067 IC50 = 0.54 nM T13127 CQ6JI3 44375143 IC50 = 4.7 nM T13127 CBOG82 44375191 IC50 = 0.8 nM T13127 CQV50W 44375199 IC50 = 3.6 nM T13127 CH2SK3 44375291 IC50 = 0.63 nM T13127 CA6GD9 44375292 IC50 = 0.37 nM T13127 CZ84FC 44375293 IC50 = 0.66 nM T13127 CGJ61P 44375312 IC50 = 25 nM T13127 C7X4FK 44375313 IC50 = 2.4 nM T13127 C45BDT 44375314 IC50 = 0.15 nM T13127 CP7D9M 44375320 IC50 = 0.12 nM T13127 CNAE75 44375332 IC50 = 0.29 nM T13127 C1Z9MS 44375398 IC50 = 2.1 nM T13127 CMH4W1 44375409 IC50 = 0.3 nM T13127 CY6W0D 44375536 IC50 = 15 nM T13127 CR8C1O 44375537 IC50 = 0.91 nM T13127 CLX9N8 44375575 IC50 = 16 nM T13127 C4BA6L 44375596 IC50 = 140 nM T13127 C7ZCM2 44375597 IC50 = 2.7 nM T13127 C7W2GU 44375614 IC50 = 0.59 nM T13127 C5RZA9 44375617 IC50 = 2.9 nM T13127 CJDW75 44375639 IC50 = 0.29 nM T13127 C6IZD1 44375709 IC50 = 1.4 nM T13127 CT0I7R 44375877 IC50 = 57 nM T13127 CE49ZQ 44377803 IC50 = 26 nM T13127 C6FDN3 44377847 IC50 = 9 nM T13127 CHYU39 44377880 IC50 = 18 nM T13127 CIAD74 44377895 IC50 = 47 nM T13127 CP84UE 44377897 IC50 = 8 nM T13127 C9DZ7J 44377898 IC50 = 22 nM T13127 C5UA4V 44377913 IC50 = 62 nM T13127 C24YKS 44377919 IC50 = 23 nM T13127 CMI8R2 44377949 IC50 = 78 nM T13127 CWC4K2 44377950 IC50 = 6 nM T13127 C8P4RG 44377956 IC50 = 32 nM T13127 C49GFJ 44377962 IC50 = 13 nM T13127 C0J6XE 44378052 IC50 = 10 nM T13127 C2E8CJ 44378053 IC50 = 6 nM T13127 CB2O6Q 44378064 IC50 = 142 nM T13127 C3D5YG 44378066 IC50 = 15 nM T13127 CJ76CQ 44378069 IC50 = 17 nM T13127 C4FOX9 44378143 IC50 = 23 nM T13127 CVZ1M5 44378154 IC50 = 15 nM T13127 CAP03Q 44378158 IC50 = 26 nM T13127 C0Z4IQ 44378159 IC50 = 55 nM T13127 CC7N9H 44378160 IC50 = 3 nM T13127 CRP60Z 44378167 IC50 = 10 nM T13127 CM6S2B 44381682 IC50 = 41 nM T13127 C12KEF 44381762 IC50 > 50000 nM T13127 CS5Y8I 44381970 IC50 = 31 nM T13127 C8A3CI 44382032 IC50 > 50000 nM T13127 C7AO4R 44382251 IC50 = 380 nM T13127 CC4S5U 44382681 IC50 = 1240 nM T13127 CUS3J4 44382757 IC50 = 1800 nM T13127 CI6DQ8 44383511 IC50 = 150 nM T13127 C6JWN8 44390085 IC50 > 10000 nM T13127 CSA3X8 44390086 IC50 > 10000 nM T13127 CLD1W8 44391495 IC50 = 3.1 nM T13127 C80GVR 44391496 IC50 = 0.9 nM T13127 C1CMU6 44391497 IC50 = 1.2 nM T13127 C8KT2M 44391501 IC50 = 7.6 nM T13127 CV4DU8 44391508 IC50 = 0.9 nM T13127 CP21RW 44391514 IC50 = 4.6 nM T13127 CX1W3J 44391515 IC50 = 4 nM T13127 C1CV5O 44391520 IC50 = 3.9 nM T13127 C3ND0P 44391522 IC50 = 0.9 nM T13127 C0B5LC 44391529 IC50 = 0.7 nM T13127 C27YUI 44391537 IC50 = 2.6 nM T13127 C0U1JA 44391539 IC50 > 5000 nM T13127 CJB3G6 44391540 IC50 = 0.9 nM T13127 CWIK23 44391544 IC50 = 3.5 nM T13127 C5XMR7 44391557 IC50 = 0.8 nM T13127 C31NER 44391563 IC50 = 48 nM T13127 C5E3AM 44391564 IC50 = 17 nM T13127 CHOK61 44391952 IC50 = 1.1 nM T13127 CN41SX 44394915 IC50 = 0.31 nM T13127 CPWC03 44394924 IC50 = 0.27 nM T13127 C6WCY4 44394934 IC50 = 0.03 nM T13127 C1UO2F 44394940 IC50 = 0.46 nM T13127 CT0K5Q 44394952 IC50 = 2.1 nM T13127 C4A9JH 44394953 IC50 = 0.37 nM T13127 CY03BF 44394963 IC50 = 1.2 nM T13127 CX2LT6 44394968 IC50 = 1.2 nM T13127 CTF0K9 44394980 IC50 = 0.36 nM T13127 CJLQ24 44394988 IC50 = 0.6 nM T13127 C7C2KJ 44394995 IC50 = 0.37 nM T13127 CK9B0V 44396117 IC50 = 16 nM T13127 CMO81D 44396157 IC50 = 3.3 nM T13127 CHE01Q 44405763 IC50 = 100 nM T13127 CTZ04C 44405819 IC50 = 70 nM T13127 CDL90A 44405831 IC50 = 30 nM T13127 C7JP9S 44405834 IC50 = 960 nM T13127 CP3WF4 44405877 IC50 = 187 nM T13127 CTG0Q1 44405882 IC50 > 1000 nM T13127 CSWA24 44405905 IC50 = 99.3 nM T13127 CQ49UZ 44406934 IC50 = 8.4 nM T13127 CY07AN 44406936 IC50 = 11 nM T13127 CGB3L8 44406942 IC50 = 9.1 nM T13127 CJ52QY 44406949 IC50 = 20 nM T13127 CKZ2N4 44406950 IC50 = 4.2 nM T13127 CPIZ82 44406952 IC50 = 49 nM T13127 C6K5IT 44406955 IC50 = 7 nM T13127 C6ZLD9 44406956 IC50 = 22 nM T13127 CLHA12 44406958 IC50 = 17 nM T13127 C0VOP1 44406959 IC50 = 21 nM T13127 CAPC35 44406963 IC50 = 59 nM T13127 C6TS9G 44406965 IC50 = 8 nM T13127 C5N8ER 44406966 IC50 = 7.9 nM T13127 CEA72D 44406967 IC50 = 11 nM T13127 CE17PN 44407015 IC50 = 20 nM T13127 C0A9CD 44407018 IC50 = 75 nM T13127 CI74ZL 44407026 IC50 = 15 nM T13127 C4RS9C 44407035 IC50 = 1800 nM T13127 C7SFL6 44407039 IC50 = 190 nM T13127 C2RH9F 44407045 IC50 = 560 nM T13127 C8IEF7 44407046 IC50 = 14 nM T13127 C2CP6S 44407047 IC50 = 9.1 nM T13127 C4LAT9 44407054 IC50 = 50 nM T13127 C7BN6A 44407061 IC50 = 490 nM T13127 CFO90Z 44407062 IC50 = 760 nM T13127 C2PL4C 44407064 IC50 = 12 nM T13127 CB9Q2U 44407068 IC50 = 5.7 nM T13127 CD8RY0 44407069 IC50 = 80 nM T13127 C4H8NZ 44407072 IC50 = 45 nM T13127 CLG8U6 44407076 IC50 = 47 nM T13127 CE2G7I 44407082 IC50 = 51 nM T13127 CJE7A6 44407090 IC50 = 13 nM T13127 C4CIG5 44407105 IC50 = 7 nM T13127 CM7E8X 44407106 IC50 = 13 nM T13127 CFT73Z 44407107 IC50 = 91 nM T13127 C6V5AE 44407148 IC50 = 12 nM T13127 CJ3W8M 44407150 IC50 = 12 nM T13127 C2DRI3 44407151 IC50 = 53 nM T13127 C1SW0B 44407155 IC50 = 28 nM T13127 C2SG1D 44407160 IC50 = 18 nM T13127 CZK2S1 44407679 IC50 = 150 nM T13127 CCTD30 44407784 IC50 = 76 nM T13127 C0D1MC 44409692 IC50 = 0.8 nM T13127 CPG97U 44409696 IC50 = 40 nM T13127 C03VQO 44409724 IC50 = 3.8 nM T13127 CPJO93 44409725 IC50 = 2.8 nM T13127 CPV54U 44409766 IC50 = 1 nM T13127 C71XNJ 44409857 IC50 = 851.14 nM T13127 C4M3TH 44409894 IC50 = 19000 nM T13127 CU58YC 44409898 IC50 = 61 nM T13127 CNQ3B8 44409901 IC50 = 2500 nM T13127 C9TV2Q 44409983 IC50 = 4.8 nM T13127 CMC0L8 44409986 IC50 = 500 nM T13127 CIA6K0 44416206 IC50 = 30 nM T13127 C14IBV 44442328 IC50 = 44.8 nM T13127 CC0LF6 44442330 IC50 = 46.5 nM T13127 CJ8P3I 44442333 IC50 = 43 nM T13127 CY4NV5 44442335 IC50 = 285 nM T13127 C7SM1U 44442338 IC50 = 45 nM T13127 CQY58L 44445070 IC50 = 0.15 nM T13127 CLP02T 44445098 IC50 = 61 nM T13127 C2RD1W 44458003 IC50 = 475 nM T13127 C0Q4LP 44458221 IC50 = 9.6 nM T13127 CNI63R 44458257 IC50 = 13 nM T13127 CCI3Y7 44458261 IC50 = 3400 nM T13127 CQYL28 44458270 IC50 = 230 nM T13127 CA68JR 44458273 IC50 = 860 nM T13127 CNQC13 44458275 IC50 = 200 nM T13127 CXR2W0 44458291 IC50 = 440 nM T13127 CI1DO9 44458817 EC50 = 6.9 nM T13127 CNO31Q 44459100 EC50 = 130 nM T13127 CI9ZK4 44459321 EC50 = 49 nM T13127 CN02QA 44459344 EC50 = 4 nM T13127 COA1V2 44459504 IC50 = 0.41 nM T13127 CEJ0K9 44459509 EC50 = 2.74 nM T13127 CL8G5A 44459510 IC50 = 0.66 nM T13127 CAD74Y 44459594 EC50 = 0.1 nM T13127 CG4LH7 44459775 EC50 = 170 nM T13127 C39TIB 44459799 EC50 = 3.8 nM T13127 C6RBS7 44459800 EC50 < 1 nM T13127 C97BTH 44459819 IC50 = 0.8 nM T13127 CF2XW7 44459847 EC50 < 1 nM T13127 C4KA0M 44459853 IC50 = 0.7 nM T13127 C7V4FJ 44459924 EC50 < 0.1 nM T13127 CCT41B 44481200 IC50 = 77 nM T13127 CU54KQ 44562318 IC50 = 67 nM T13127 CT7A4P 44564603 IC50 = 6.3 nM T13127 C8P5GE 44564604 IC50 = 4 nM T13127 CH7SJ5 44564605 IC50 = 3.4 nM T13127 CGT4B6 44564606 IC50 = 0.7 nM T13127 CZ57ED 44564619 IC50 = 170 nM T13127 C52LPR 44564620 IC50 = 360 nM T13127 CHM57T 44564621 IC50 = 360 nM T13127 C4BZ0X 44564622 IC50 > 1000 nM T13127 CC98DF 44564623 IC50 = 7.2 nM T13127 CW5RH1 44564624 IC50 = 3.2 nM T13127 CCAF82 44564625 IC50 = 0.9 nM T13127 CIXH71 44564626 IC50 = 2 nM T13127 CJU2K4 44564916 IC50 = 850 nM T13127 CZ5NM8 44564917 IC50 = 30 nM T13127 C0CRU5 44564918 IC50 = 250 nM T13127 C4BFQ7 44564960 IC50 = 3.3 nM T13127 C2V7IR 44564961 IC50 = 8.5 nM T13127 CJ31NT 44564962 IC50 = 2.8 nM T13127 CMF4V1 44564963 IC50 = 11 nM T13127 CA3BE9 44564964 IC50 = 1 nM T13127 CVC8P0 44564965 IC50 = 11 nM T13127 C4YS2E 44564966 IC50 = 2.6 nM T13127 C3ROU2 44564967 IC50 = 6.4 nM T13127 CV2NU6 44564968 IC50 = 2.4 nM T13127 CCL0A1 44565020 IC50 = 1.5 nM T13127 CVLT23 44565021 IC50 = 49 nM T13127 C8I4DV 44565022 IC50 = 0.8 nM T13127 CR4XW9 44565023 IC50 = 1.2 nM T13127 C2U5KV 44593866 IC50 = 0.3 nM T13127 CH67TX 45484000 IC50 > 50000 nM T13127 C7AT3B 45484001 IC50 = 450 nM T13127 CZB4V7 46230597 IC50 = 130000 nM T13127 CX8OF9 46230598 IC50 = 160000 nM T13127 C8XZL4 46230599 IC50 = 60000 nM T13127 CC13OA 46230630 IC50 > 200000 nM T13127 CM82AY 46230631 IC50 = 60000 nM T13127 CB27VP 46230633 Ki = 260 nM T13127 C3SQ4F 46230634 IC50 = 10000 nM T13127 CVN05P 46230681 IC50 = 60000 nM T13127 CFIX74 46230683 IC50 > 200000 nM T13127 CM8DU9 46230685 IC50 = 85000 nM T13127 CYU16M 46230686 IC50 > 200000 nM T13127 CAW9N8 46230688 Ki = 500 nM T13127 CG1RA3 46230690 Ki = 230 nM T13127 C4TJ6C 46230733 IC50 = 21000 nM T13127 CLE52I 46230735 IC50 = 12000 nM T13127 CRK6N4 46231898 IC50 = 12 nM T13127 CH3JZ9 49781429 IC50 = 5400 nM T13127 CBR29D 49781430 IC50 > 10000 nM T13127 C2DW9S 49781656 IC50 = 5300 nM T13127 CG4DJ5 49781657 IC50 = 6850 nM T13127 C4PY6Q 49781661 IC50 = 48 nM T13127 CDB12N 49781870 IC50 = 85 nM T13127 CUMR38 49782332 IC50 = 550 nM T13127 C5RP3L 49782333 IC50 = 520 nM T13127 CW17AZ 49782546 IC50 = 110 nM T13127 CC25UW 49782547 IC50 = 620 nM T13127 CX0PS3 49782548 IC50 = 230 nM T13127 CUFV75 49782549 IC50 = 64 nM T13127 C6NZ1R 49782773 IC50 = 290 nM T13127 CEW47F 49782774 IC50 = 490 nM T13127 C2O6LW 49782775 IC50 = 320 nM T13127 CFMK50 49782776 IC50 = 870 nM T13127 CW2X5H 49782980 IC50 = 2300 nM T13127 C0F6CW 49782981 IC50 = 510 nM T13127 CH0BI7 49782982 IC50 = 6200 nM T13127 CJ2H3X 49782984 IC50 = 590 nM T13127 CFV08K 49783194 IC50 = 400 nM T13127 C2V4GL 49783195 IC50 = 250 nM T13127 C8GC2J 49783396 IC50 = 350 nM T13127 CB0T1G 49799946 IC50 = 1.1 nM T13127 CQS80F 49859768 IC50 = 2.8 nM T13127 CN0GM9 49863899 IC50 = 4340 nM T13127 CVL4N1 51356543 Ki = 5 nM T13127 CG90UM 52940843 IC50 = 5300 nM T13127 C1IX7S 52943729 IC50 = 720 nM T13127 C0QBI4 53317632 IC50 = 14700 nM T13127 CA2TZ5 53317633 IC50 > 100000 nM T13127 C2I4VM 53320241 IC50 > 100000 nM T13127 C52BPN 53321567 IC50 > 100000 nM T13127 C1CPK9 53322673 IC50 > 100000 nM T13127 C1H8WU 53322894 IC50 > 100000 nM T13127 CWK84N 53324228 IC50 > 100000 nM T13127 CS5H8U 53326789 IC50 > 100000 nM T13127 CL8ZP9 53709990 IC50 = 9000 nM T13127 C0IZW6 54763547 IC50 = 1200 nM T13127 CC5K7H 56657726 IC50 = 1.8 nM T13127 C2Z1AE 56657870 IC50 = 110 nM T13127 CWZ08N 56661382 IC50 = 1400 nM T13127 CW7DU4 56664851 IC50 = 1.2 nM T13127 C9JZ8R 56664853 IC50 = 2.2 nM T13127 C9UPY5 56668261 IC50 = 25 nM T13127 CJ14CL 56671724 IC50 = 21 nM T13127 CZ45SG 56675152 IC50 = 0.123 nM T13127 CDLN19 56675153 IC50 = 30 nM T13127 CI0WH4 56675646 IC50 = 90000 nM T13127 C4LPB8 56678448 IC50 = 42 nM T13127 CWB8T6 56681790 IC50 = 1600 nM T13127 CKF59V 56681791 IC50 = 4.8 nM T13127 C2UKS0 59122512 IC50 = 0.6 nM T13127 CS8I0G 59122517 IC50 = 0.7 nM T13127 CUH6F9 59122522 IC50 = 1.4 nM T13127 C4VB1G 59122524 IC50 = 0.6 nM T13127 CAX7S3 59122525 IC50 = 1.4 nM T13127 CVOM93 59122527 IC50 = 5.5 nM T13127 CU98HF 59122528 IC50 = 2.6 nM T13127 C17SCO 59122530 IC50 = 0.9 nM T13127 CUY84A 59122532 IC50 = 0.2 nM T13127 C1M6DC 59122534 IC50 = 0.6 nM T13127 C3FRG7 59122535 IC50 = 0.4 nM T13127 CW3JB7 59122545 IC50 = 0.1 nM T13127 C8I5KF 59122547 IC50 = 1.7 nM T13127 CAC1E3 59122579 IC50 = 1.8 nM T13127 C4WL7H 59122626 IC50 = 5 nM T13127 CDH7A6 59122650 IC50 > 18 nM T13127 C6EMA3 70684027 IC50 = 5200 nM T13127 C6A7DT 70684028 IC50 = 1300 nM T13127 C3Q2BG 70688302 IC50 = 8300 nM T13127 CDV6A1 70690305 IC50 = 7700 nM T13127 C41ZVQ 70692484 IC50 = 24300 nM T13127 C39FKV 70694520 IC50 = 1500 nM T13127 C1KX2T 70697542 IC50 > 100000 nM T13127 C9HCE0 71356515 IC50 = 19700 nM T13127 CZ0A5R 71450984 IC50 = 14000 nM T13127 CHM04F 71451486 IC50 = 3350 nM T13127 CY4Q0V 71452753 IC50 = 3400 nM T13127 CS51JP 71459970 IC50 = 33 nM T13127 C9RYU1 71460517 IC50 = 17210 nM T13127 CDC2T7 71462437 IC50 > 9700 nM T13127 C5Q3XG 71521669 IC50 > 500000 nM T13127 C7LSP6 71522036 IC50 = 39000 nM T13127 CZGD29 71569242 IC50 = 43090 nM T13127 C4F3XW 71569891 IC50 = 650 nM T13127 CNTQ52 71569892 IC50 = 630 nM T13127 C0BMR2 71569893 IC50 = 1200 nM T13127 CV4U1L 71569894 IC50 = 1070 nM T13127 CBQ04R 71716101 IC50 = 4920 nM T13127 CSY3A0 71716102 IC50 = 13100 nM T13127 CO5QD7 71716103 IC50 = 10980 nM T13127 C3O1TL 71716108 IC50 = 4670 nM T13127 CND1I8 71716109 IC50 = 5330 nM T13127 CJDU78 71716727 IC50 = 10290 nM T13127 CEN39B 71717921 IC50 = 14980 nM T13127 C82DAE 71718541 IC50 = 13740 nM T13127 C2AK7Q 71718546 IC50 = 86490 nM T13127 C6DU4H 71718590 IC50 = 400000 nM T13127 CO8D3U 71719145 IC50 = 3180 nM T13127 CD8C3A 71719146 IC50 = 7270 nM T13127 CV82MQ 71719753 IC50 = 7010 nM T13127 C20DNR 71719754 IC50 = 6360 nM T13127 CS9DZ7 71723295 Ki = 837 nM T13127 C01ZOP 73351357 IC50 = 500000 nM T13127 CWBT35 76310611 IC50 > 18 nM T13127 C4ULX7 76311224 IC50 = 1700 nM T13127 CJ75FT 76311225 IC50 = 9300 nM T13127 CA7IL6 76311226 IC50 = 3700 nM T13127 CY0F7A 76311227 IC50 > 50000 nM T13127 C5E7FI 76311228 IC50 = 5600 nM T13127 C5WJ9V 76311229 IC50 = 10400 nM T13127 C3D2OT 76314839 IC50 = 1100 nM T13127 CHFV59 76314840 IC50 = 4700 nM T13127 C9LS3T 76317816 IC50 > 20 nM T13127 C2DBJ1 76318444 IC50 > 50000 nM T13127 CY3AV6 76321526 IC50 = 1.9 nM T13127 CV52HT 76322113 IC50 = 48.9 nM T13127 CVB76L 76322114 IC50 = 1460 nM T13127 CI89QS 76322115 IC50 = 24000 nM T13127 CS41ZO 76325137 IC50 = 3.2 nM T13127 CUL89Z 76325138 IC50 = 3.2 nM T13127 C8IBO3 76325733 IC50 = 460 nM T13127 CKV31J 76325734 IC50 = 1900 nM T13127 CM4VE9 76325736 IC50 = 140 nM T13127 CD12RZ 76325737 IC50 = 1900 nM T13127 C9UJN7 76327916 IC50 = 7000 nM T13127 CXD97F 76328691 IC50 = 1.8 nM T13127 CQ2R4D 76329303 IC50 = 140 nM T13127 C1DBY3 76329304 IC50 > 50000 nM T13127 CF21NJ 76329305 IC50 = 21600 nM T13127 CG0J2R 76329306 IC50 = 42 nM T13127 CHS6R7 76329307 IC50 > 50000 nM T13127 C2E4LY 76329308 IC50 = 67 nM T13127 C2NFE0 76332951 IC50 = 1800 nM T13127 C8U0PI 76332952 IC50 = 23000 nM T13127 CP5Z2F 76332953 IC50 = 8700 nM T13127 C4Q2FI 76335995 IC50 = 0.8 nM T13127 C8X3IS 76335996 IC50 = 0.1 nM T13127 CKJ30N 76336563 IC50 = 3520 nM T13127 CI59ZC 76336564 IC50 > 50000 nM T13127 CNV47W 76336565 IC50 = 76 nM T13127 C8MCZ7 76901065 IC50 = 15 nM T13127 CML51R 76901066 IC50 = 2270 nM T13127 C5M0WH 76901067 IC50 = 7.2 nM T13127 C3MHW0 76901249 IC50 = 32 nM T13127 C72TUG 76901250 IC50 = 13 nM T13127 C3STE0 76901251 IC50 = 9.6 nM T13127 CUKC42 76901252 IC50 = 71 nM T13127 COM8C7 76901253 IC50 = 910 nM T13127 C0Z2IB 76901436 IC50 = 580 nM T13127 CEZ1F7 76901437 IC50 = 17 nM T13127 C92ADI 76901438 IC50 = 23 nM T13127 C6QPY5 76901439 IC50 = 1940 nM T13127 C13PKQ 76901440 IC50 = 2.9 nM T13127 C64GIJ 76901621 IC50 = 450 nM T13127 CCN1G9 76901623 IC50 = 710 nM T13127 CLF4S1 76901624 IC50 = 38 nM T13127 CF9EM3 89267667 IC50 = 41 nM T13127 CP9LX7 90656272 IC50 = 400000 nM T13127 C07IKQ 90656274 IC50 = 340000 nM T13127 CU0T9S 90665658 IC50 = 1.35 nM T13127 CAE45N 90665659 IC50 > 50000 nM T13127 C1W2SC 90665660 IC50 = 1.8 nM T13127 C02BZU 90667612 IC50 > 50000 nM T13127 C6AQ3V 90667613 IC50 = 9900 nM T13127 CQ4RH5 90667614 IC50 = 19000 nM T13127 CQG4S8 90667615 IC50 > 50000 nM T13127 CR7AM6 90667616 IC50 = 29000 nM T13127 CTY2L9 90667617 IC50 = 9200 nM T13127 C3OVP0 90667618 IC50 = 25000 nM T13127 CX5HD7 90667620 IC50 > 50000 nM T13127 C56LBD 90667621 IC50 > 50000 nM T13127 CQC3G2 90667622 IC50 = 29000 nM T13127 CS3Q5M 90667623 IC50 = 36000 nM T13127 CXCV73 90667624 IC50 > 50000 nM T13127 CENJ02 90667625 IC50 = 3900 nM T13127 CV5XP2 90667626 IC50 = 11000 nM T13127 CA1CE2 90667627 IC50 = 18000 nM T13127 CU6Y7V 90667628 IC50 > 50000 nM T13127 CC9FU3 90667629 IC50 = 2700 nM T13127 CQ36NC 90667630 IC50 = 5000 nM T13127 CP4G3X 90667631 IC50 = 34000 nM T13127 CXGE97 90667632 IC50 > 50000 nM T13127 C0UK6E 90667633 IC50 = 5900 nM T13127 CCK2N9 90667634 IC50 = 40000 nM T13127 CEF4A1 90667635 IC50 > 50000 nM T13127 CMV40T 90667636 IC50 > 50000 nM T13127 CP42WT 90667637 IC50 = 7700 nM T13127 CX52HA 90667638 IC50 = 8300 nM T13127 CR5O2Y 90667639 IC50 = 25000 nM T13127 COAG06 90667640 IC50 = 7800 nM T13127 C3IZ2D 90667641 IC50 = 14000 nM T13127 C67DMR 90667642 IC50 = 6500 nM T13127 C8R9IO 90667643 IC50 = 4000 nM T13127 CHU7E5 90667644 IC50 = 18000 nM T13127 CZO56H 90667645 IC50 > 50000 nM T13127 C7M8CY 90667648 IC50 = 27000 nM T13127 CFJ5B1 90667650 IC50 = 21000 nM T13127 CZX52C 90680670 IC50 = 5000 nM T13127 CS0U4J 90680678 IC50 = 2800 nM T13127 CB1SX0 118724655 IC50 = 20700 nM T13127 CG8V2D 118724656 IC50 = 19400 nM T13127 CC0IP2 118724658 IC50 = 32200 nM T13127 CT65ER 118724659 IC50 = 14800 nM T13127 CR0MT1 118724660 IC50 = 72300 nM T13127 CKT86L 118724663 IC50 = 22100 nM T13127 C1ZWD8 118724664 IC50 = 5900 nM T13127 C7UW5L 118724665 IC50 = 4400 nM T13127 CRGN42 118724666 IC50 = 57800 nM T13127 CN53YO 118724667 IC50 = 14900 nM T13127 CS6FY4 118724668 IC50 = 11400 nM T13127 C8T9WE 118724669 IC50 = 15300 nM T13127 C6Z0BL 118724670 IC50 = 14400 nM T13127 CVLN04 118724672 IC50 = 20800 nM T13127 COGR34 118724673 IC50 = 2600 nM T13127 CNE69T 118724674 IC50 = 1300 nM T13127 CQ4X2G 118724680 IC50 = 7300 nM T13127 CGNW92 118724681 IC50 = 20700 nM T13127 CZ2V3E 118724682 IC50 = 2200 nM T13127 CN43AS 122192720 IC50 = 65400 nM T13127 CYM07Z 122192721 IC50 = 4700 nM T13127 C9X4GY 122192722 IC50 = 40200 nM T13127 CFCH64 122192723 IC50 = 11700 nM T13127 CI1A0R 122192725 IC50 = 12000 nM T13127 CT1Y4I 122192727 IC50 = 44700 nM T13127 C0AJ5Y 122192728 IC50 = 18900 nM T13127 CEXM61 122192739 IC50 = 35000 nM T13127 CE2TO9 122194646 IC50 = 150 nM T13127 C2I6WZ 122194647 IC50 = 240 nM T13127 C8WPL7 122196006 IC50 = 27 nM T13127 C2TF4X 122196007 IC50 = 7100 nM T13127 CM3V8R 127025895 IC50 = 34000 nM T13127 CFTX92 127025896 IC50 = 290 nM T13127 CHN2T5 127025897 IC50 = 2100 nM T13127 CHWD41 127026183 IC50 = 330 nM T13127 C7JD0X 127026184 IC50 = 640 nM T13127 CQY96J 127029311 IC50 = 130 nM T13127 C1A6FB 127029312 IC50 = 190 nM T13127 C37VST 127038565 IC50 = 10 nM T13127 CU8S2K 127038918 IC50 = 980 nM T13127 CP5D4U 127039232 IC50 = 380 nM T13127 CJ0U7E 127039233 IC50 = 370 nM T13127 CI0HE2 127039234 IC50 = 5100 nM T13127 C9J4ZY 127040236 IC50 = 3600 nM T13127 CG61DY 127040237 IC50 = 1200 nM T13127 CX6Y8A 127040238 IC50 = 4600 nM T13127 CFM7X8 127040862 IC50 = 13 nM T13127 CCKM82 127040863 IC50 > 100000 nM T13127 C70YPZ 127041227 IC50 = 680 nM T13127 C3YX2F 127041228 IC50 = 150 nM T13127 CZX31V 127042110 IC50 = 970 nM T13127 CCE08O 127042111 IC50 = 22000 nM T13127 C2Q9JX 127043146 IC50 = 8740 nM T13127 C9KJ6Z 127043148 IC50 = 1320 nM T13127 C46PBD 127043149 IC50 = 9 nM T13127 CB6E7S 127043150 IC50 = 23 nM T13127 CGZA21 127043155 IC50 = 155 nM T13127 CT63IZ 127043156 IC50 = 711 nM T13127 CE0L2W 127043328 IC50 = 11630 nM T13127 C0D5ZL 127043329 IC50 = 15890 nM T13127 C03GSO 127043330 IC50 = 726 nM T13127 C7AN8Z 127043331 IC50 = 931 nM T13127 CRU05N 127043507 IC50 = 19280 nM T13127 CKZ9D1 127044461 IC50 = 2330 nM T13127 C3CO0R 127045623 IC50 = 602 nM T13127 CX0D7V 136219359 IC50 = 19690 nM T13127 C7X8HL 136219361 IC50 = 23850 nM T13127 C7WR0U 136219363 IC50 = 15560 nM T13127 CA9VZ8 136219365 IC50 = 27390 nM T13127 CIS35W 136224236 IC50 = 520 nM T13127 CA87SG 136229773 IC50 = 3730 nM T13127 CT3ON8 136239386 IC50 = 14470 nM T13127 CU81TE 136239388 IC50 = 31890 nM T13127 CH0QW4 136239390 IC50 = 22190 nM T13127 C1MUN4 136239394 IC50 = 27340 nM T13127 C2B0FY 136239501 IC50 = 20130 nM T13127 C6FYG0 136244505 IC50 = 23570 nM T13127 CJ7WF5 136244591 IC50 = 4670 nM T13127 CTIM53 136244593 IC50 = 46190 nM T13127 CS0HI9 136244595 IC50 = 43640 nM T13127 CGO0H5 136244597 IC50 = 62300 nM T13127 CQV4D1 136244599 IC50 = 12490 nM T13127 CEZ78V 136244601 IC50 = 43480 nM T13127 C6KYZ3 136254450 IC50 = 36370 nM T13127 CGBZ45 136254452 IC50 = 46190 nM T13127 C7FTV4 136254454 IC50 = 25850 nM T13127 CVI2W4 136254456 IC50 = 55220 nM T13127 CSK9C1 136254458 IC50 = 20840 nM T13127 C9KZR3 136260480 IC50 = 30940 nM T13127 CN86QX 136260482 IC50 = 48000 nM T13127 CI46HD 136260539 IC50 = 62670 nM T13127 CAG1L6 136260541 IC50 = 28230 nM T13127 COG57C 136260545 IC50 = 31360 nM T13127 CD7L2U 145982147 IC50 = 860 nM T13127 C0Q5ZF 155543825 IC50 = 0.06 nM T13127 D01OFD 10102380 IC50 = 230 nM T13127 D02FVV 370346 IC50 = 930 nM T13127 D02KVR 10099206 IC50 = 0.8 nM T13127 D06DSE 9919495 IC50 = 10 nM T13127 D06JMV 11271978 IC50 = 3.8 nM T13127 D0DM6F 11761968 EC50 = 0.18 nM T13127 D0M5PB 395754 IC50 = 0.5 nM T13127 D0PK8Y 9806149 IC50 = 0.7 nM T13127 D0R3PD 10005132 IC50 = 8000 nM T13127 D0T2SJ 23646371 IC50 = 0.3 nM T13127 D0VD2C 3037595 IC50 = 175 nM T13127 D0WT6A 3301 IC50 = 15500000 nM T13127 D0X5KQ 44320675 IC50 = 1200 nM T07533 CC48GB 9805990 IC50 = 270 nM T07533 C03LMO 9851010 IC50 = 2.6 nM T07533 C2MJB3 9869236 IC50 = 6.4 nM T07533 CGS38K 9891662 IC50 = 8.8 nM T07533 C7OXU6 9893362 IC50 = 1.3 nM T07533 C95CAK 9893401 IC50 = 43 nM T07533 CGQ63J 9912755 IC50 = 60 nM T07533 CO7JL9 10874540 IC50 = 5 nM T07533 CNQ27P 10875045 IC50 = 3 nM T07533 C3P9FZ 10895442 IC50 = 8.3 nM T07533 CC4SR0 10896240 IC50 = 1.8 nM T07533 C0GRI1 10896496 IC50 = 2.4 nM T07533 CRA54I 10917146 IC50 = 120 nM T07533 C57WJA 10918532 IC50 = 42 nM T07533 C6MJ3O 10928783 IC50 = 16 nM T07533 CK4O9I 10939283 IC50 = 8.7 nM T07533 CM9VK6 10939852 IC50 = 340 nM T07533 CYU20M 10940136 IC50 = 5.5 nM T07533 C1IZR8 10951208 IC50 = 1.7 nM T07533 CVW5R3 10961434 IC50 = 5.2 nM T07533 CAHR01 10962353 IC50 = 2.4 nM T07533 CG8WC0 10962509 IC50 = 2 nM T07533 C62AUC 10973085 IC50 = 2.2 nM T07533 C1E3HD 10973138 IC50 = 1.2 nM T07533 CY7QP0 10983506 IC50 = 120 nM T07533 CN95OR 10983704 IC50 = 2.5 nM T07533 C96UMN 10994667 IC50 = 1.6 nM T07533 CN4QG3 10994772 IC50 = 1.4 nM T07533 COP90M 10995108 IC50 = 1.8 nM T07533 CIL7D4 10995390 IC50 = 1 nM T07533 C21TIL 11004943 IC50 = 6.6 nM T07533 C61DIZ 11027521 IC50 = 6.5 nM T07533 CX0I1A 11027680 IC50 = 2.3 nM T07533 CFVH36 11049142 IC50 = 1.1 nM T07533 CNE1M2 11123287 IC50 = 1.9 nM T07533 CQJR21 11124756 IC50 = 1.6 nM T07533 CSC8O9 11145136 IC50 = 15 nM T07533 CQEA84 11145472 IC50 = 10 nM T07533 C4W1DI 11730355 IC50 = 12 nM T07533 CA9L4W 11733571 IC50 = 4.1 nM T07533 CLID72 11734494 IC50 = 1.9 nM T07533 C4LRQ2 11762346 IC50 = 2 nM T07533 CL4BI2 11762419 IC50 = 0.7 nM T07533 CQ9JC1 11827152 IC50 = 2.5 nM T07533 C1HO2U 44361523 IC50 = 2.2 nM T07533 CDZ19W 44361568 IC50 = 3.4 nM T07533 CBR57W 44361595 IC50 = 0.9 nM T07533 C4HPJ2 44361825 IC50 = 7.5 nM T07533 CHA20L 44361826 IC50 = 1.8 nM T59056 D02STN 132971 IC50 = 1750 nM T59056 D02YPG 667484 IC50 = 1.7 nM T59056 D07ABV 468595 IC50 = 21 nM T59056 D09LNI 3365 IC50 = 13000 nM T59056 D0C1WH 3902 IC50 = 1420 nM T59056 D0Q9JT 4174 IC50 = 42 nM T59056 D0ZX1P 59693 IC50 = 0.8 nM T59056 D03AJU 44139752 IC50 = 0.2 nM T59056 D0E3TC 44259 IC50 = 11 nM T59056 C9LCD8 3823 IC50 = 67 nM T59056 CFO8Y3 83332 IC50 = 145 nM T59056 C5WUK4 256446 IC50 = 6 nM T59056 C78IXN 563347 IC50 = 865 nM T59056 CNG05O 571156 IC50 = 262 nM T59056 C5NT4U 583968 IC50 = 30 nM T59056 C1Y5HM 603115 IC50 = 104 nM T59056 C8HZL4 618231 IC50 = 11 nM T59056 C7XD4N 706178 IC50 = 65 nM T59056 CJ4FE1 853038 IC50 = 107 nM T59056 CI16RF 867617 IC50 = 520 nM T59056 CC29WP 886929 IC50 = 309 nM T59056 C6S1WJ 955210 IC50 > 1000 nM T59056 CB5KN2 1118253 IC50 = 82 nM T59056 CB8QN3 1214447 IC50 = 7 nM T59056 C7LS3G 1515242 IC50 = 40 nM T59056 CB93KS 1550302 IC50 < 10000 nM T59056 C83OBD 3021561 IC50 = 411 nM T59056 CBY4W2 3102914 IC50 > 1000 nM T59056 CBF75X 5376779 IC50 < 10000 nM T59056 C7VSM2 5702471 IC50 = 12000 nM T59056 CST49O 5702960 IC50 < 10000 nM T59056 C1JAT6 6539761 IC50 = 22 nM T59056 CTE57C 6539762 IC50 = 141 nM T59056 CF17BE 6539771 IC50 = 57 nM T59056 CJ7RS8 6539772 IC50 = 878 nM T59056 CQD13Z 6539787 IC50 = 15 nM T59056 CQB1U5 6539798 IC50 = 22 nM T59056 C79FTC 6539799 IC50 = 56 nM T59056 C5Z9KY 6539802 IC50 = 11 nM T59056 C7CAB8 6539809 IC50 = 14 nM T59056 COU5D2 6539810 IC50 = 31 nM T59056 CQ0HD5 6539812 IC50 = 57 nM T59056 CQ9XM0 6539813 IC50 = 65 nM T59056 CF1R9J 6539815 IC50 = 20 nM T59056 CMA37K 6539816 IC50 = 14 nM T59056 CP4VI2 6540030 IC50 = 24.8 nM T59056 CR6LS8 6540031 IC50 = 9.6 nM T59056 CU3C1Y 6540034 IC50 = 22.7 nM T59056 CXEW82 6540035 IC50 = 35.9 nM T59056 CBKX32 6540037 IC50 = 47.3 nM T59056 C8MRI7 6540038 IC50 = 16.7 nM T59056 C8JXY1 6540039 IC50 = 13.9 nM T59056 CZK3T4 6540040 IC50 = 88.8 nM T59056 CDS26H 6540041 IC50 = 3.7 nM T59056 CG13VT 6540057 IC50 = 45 nM T59056 C75OWB 6540058 IC50 = 448 nM T59056 CG9RF6 7515053 IC50 < 10000 nM T59056 C2BUR8 9837726 IC50 = 50 nM T59056 CX38PV 9927427 IC50 = 40 nM T59056 C49HDL 10013868 IC50 = 73000 nM T59056 C5NAU2 10036028 IC50 = 90000 nM T59056 C3YC9I 10263082 IC50 = 59 nM T59056 CTUL01 10331100 IC50 = 55000 nM T59056 CYNM04 10376335 IC50 = 43000 nM T59056 CP8G9A 10398594 IC50 = 24000 nM T59056 CH7IA3 10489983 IC50 = 10000 nM T59056 CG0A6X 10513321 IC50 = 20000 nM T59056 CTH96I 10584844 IC50 = 30 nM T59056 CN2RF5 10585362 IC50 < 10000 nM T59056 CTI0R2 10587179 IC50 < 10000 nM T59056 CZ2H3N 10610950 IC50 < 10000 nM T59056 C04DNA 10656613 IC50 < 10000 nM T59056 CA13SW 10711620 IC50 = 124 nM T59056 CO3JR0 10727176 IC50 = 19000 nM T59056 CBG72H 10729611 IC50 < 10000 nM T59056 CFE87L 10729612 IC50 < 10000 nM T59056 CHL74J 10752290 IC50 < 10000 nM T59056 CM3GX1 10753431 IC50 < 10000 nM T59056 CG27MD 10776192 IC50 = 21000 nM T59056 CNGQ30 10800145 IC50 < 10000 nM T59056 CZW6V4 10828130 IC50 = 19.5 nM T59056 CW0L6P 11021023 IC50 = 41 nM T59056 C6G3JV 11032034 IC50 = 7 nM T59056 C1TP7W 11232831 IC50 = 289 nM T59056 C58MTC 11543201 IC50 > 500 nM T59056 CN4T0K 11544009 IC50 = 28 nM T59056 C9IJ3T 11594132 IC50 = 72 nM T59056 CZ50DQ 11708478 IC50 = 68 nM T59056 CW2B3A 11738647 IC50 = 2190 nM T59056 C27WEU 12229396 IC50 = 637 nM T59056 CCU19N 13045366 IC50 = 62 nM T59056 C4ELY3 13276694 IC50 = 60 nM T59056 C1F5IT 13688212 IC50 = 40 nM T59056 C8WU6R 14424120 IC50 > 1000 nM T59056 C0C4JN 15591368 IC50 = 3 nM T59056 CQ03PZ 16654684 IC50 > 1000 nM T59056 C4ZVL5 16752765 IC50 = 3 nM T59056 CY0RV3 18668566 IC50 = 39 nM T59056 CRDM03 18679298 IC50 = 110 nM T59056 CN8IQ3 18785133 IC50 = 3.467 nM T59056 C1R2FU 22406650 IC50 = 499.5 nM T59056 C6D2NZ 24692916 IC50 = 1000 nM T59056 C07XJP 24696760 IC50 = 78 nM T59056 CW3C5U 24896569 IC50 = 11 nM T59056 C29WQM 25033651 IC50 = 436 nM T59056 C1VPF8 25033652 IC50 = 1676 nM T59056 C9Q8ZK 25033657 IC50 = 311 nM T59056 CWIC10 25033659 IC50 = 1492 nM T59056 CAI47X 25033725 IC50 = 518 nM T59056 CW5A1U 25033730 IC50 = 840 nM T59056 CV49HP 25033731 IC50 = 945 nM T59056 C86AIT 25033734 IC50 = 121 nM T59056 CEJ89P 25033804 IC50 = 991 nM T59056 C3UF1V 25033806 IC50 = 543 nM T59056 CF46OB 25033808 IC50 = 567 nM T59056 CBI59C 25033810 IC50 = 587 nM T59056 CV19DG 25034278 IC50 = 4.5 nM T59056 CEP93C 25034345 IC50 = 1.2 nM T59056 CSX16E 25034347 IC50 = 0.8 nM T59056 CXDF80 25034348 IC50 = 2.1 nM T59056 C56WJS 25034349 IC50 = 6.9 nM T59056 CGD93B 25034350 IC50 = 9.1 nM T59056 CK3L1J 25034351 IC50 = 22 nM T59056 C9MF8O 25034425 IC50 = 0.5 nM T59056 CW7V9I 25034428 IC50 = 0.5 nM T59056 CH6U1E 25034429 IC50 = 3.3 nM T59056 CLP17I 25034432 IC50 = 3.8 nM T59056 CTB95M 25034489 IC50 = 94 nM T59056 CBLS47 25034490 IC50 = 1216 nM T59056 CW82MN 25034491 IC50 = 0.2 nM T59056 CJ8M0E 25034492 IC50 = 2.2 nM T59056 COSJ63 25034493 IC50 = 0.2 nM T59056 C7KAR1 25034657 IC50 = 816 nM T59056 C0MEI5 25129119 IC50 = 2.7 nM T59056 C2QU1N 25129120 IC50 = 3.9 nM T59056 C2FE6G 25129122 IC50 = 7.6 nM T59056 CJ48LA 25129123 IC50 = 3 nM T59056 CX4GM7 25129462 IC50 = 119 nM T59056 C9IFV2 25129463 IC50 = 65 nM T59056 C6D8UQ 25129464 IC50 = 28 nM T59056 CJCE15 25130854 IC50 = 7.7 nM T59056 C9AS7H 25131165 IC50 = 24 nM T59056 C9G8MJ 25131494 IC50 = 5 nM T59056 CA7OP2 25131495 IC50 = 30 nM T59056 C1WM2B 25147691 IC50 = 0.1 nM T59056 CYT15G 25180102 IC50 = 101 nM T59056 CGX76Y 25180105 IC50 = 30 nM T59056 CMU54R 25180107 IC50 = 1.6 nM T59056 C0XHA2 25180109 IC50 = 2.6 nM T59056 C9LQJ6 25180110 IC50 = 22 nM T59056 CHJ2S3 25180298 IC50 = 2.7 nM T59056 C1HGB6 25180299 IC50 = 3.8 nM T59056 C90UKD 25180304 IC50 = 3.3 nM T59056 CPQ6A9 25180305 IC50 = 5.1 nM T59056 C6ZE9H 25180500 IC50 = 1.8 nM T59056 C6FN2Z 25180502 IC50 = 64 nM T59056 C9DB1G 25180503 IC50 = 0.2 nM T59056 CIZ82U 25180504 IC50 = 4.2 nM T59056 CJS97E 30507078 IC50 = 53.5 nM T59056 CHI5Y2 39231360 IC50 > 1000 nM T59056 C70VMZ 44203017 IC50 > 10000 nM T59056 CT3XM4 44206480 IC50 = 15.85 nM T59056 C9UWB5 44206481 IC50 = 3.981 nM T59056 C1I0NW 44381001 IC50 = 14000 nM T59056 CDTS58 44387709 IC50 = 35.7 nM T59056 CT4L0R 44455927 IC50 = 277 nM T59056 C69QUY 44456068 IC50 > 1000 nM T59056 CM8BT1 44456104 IC50 = 3407 nM T59056 C68FJH 44456188 IC50 = 4391 nM T59056 CP50NM 44456189 IC50 = 1665 nM T59056 CVR70K 44456190 IC50 > 1000 nM T59056 C9JCL1 44456223 IC50 = 2153 nM T59056 C6BE0T 44456226 IC50 = 1423 nM T59056 CO4PI7 44479388 IC50 = 1.1 nM T59056 C1K6QY 44479389 IC50 = 2.4 nM T59056 CLPH49 44479390 IC50 = 0.6 nM T59056 C2EM5N 44479391 IC50 = 0.2 nM T59056 CNTI30 44479392 IC50 = 0.9 nM T59056 C40IPE 44479393 IC50 = 0.2 nM T59056 C8JHS9 44479641 IC50 = 1.2 nM T59056 C2P4XT 44479643 IC50 = 1 nM T59056 CWP4Y8 44479644 IC50 = 5.9 nM T59056 C81QJE 44479645 IC50 = 4.4 nM T59056 CO8T3N 44479646 IC50 = 89 nM T59056 C4YN0S 44479648 IC50 = 56 nM T59056 CF12OV 44479882 IC50 = 1.3 nM T59056 CCN58W 44479883 IC50 = 2.2 nM T59056 C7GV6X 44479884 IC50 = 15 nM T59056 CH8RO1 44479885 IC50 = 0.9 nM T59056 CES96D 44479886 IC50 = 1.4 nM T59056 CH02ZN 44480128 IC50 = 1.4 nM T59056 C1LSH2 44480129 IC50 = 4.6 nM T59056 C3UQS0 44480130 IC50 = 0.7 nM T59056 C4KG5O 44480131 IC50 = 33 nM T59056 COI7E8 44480132 IC50 = 2.3 nM T59056 C9KS5O 44480133 IC50 = 16 nM T59056 CLMI41 44480134 IC50 = 2.4 nM T59056 CYH9A6 44480385 IC50 = 41 nM T59056 C9V8CH 44480386 IC50 = 0.5 nM T59056 CL8KQ3 44480387 IC50 = 1.1 nM T59056 CT50NZ 44480388 IC50 = 89 nM T59056 CKO4N3 44480389 IC50 = 24 nM T59056 CT3MO9 44480390 IC50 = 0.3 nM T59056 CN7LT2 44482245 IC50 = 11 nM T59056 CO63LK 44569291 IC50 = 187 nM T59056 CW06BV 45103704 IC50 = 50 nM T59056 C9Z4YB 45103705 IC50 = 177 nM T59056 CB2FC9 45103804 IC50 = 120.23 nM T59056 C4Q2FU 45103806 IC50 = 54.95 nM T59056 CQF56Z 45103807 IC50 = 58.88 nM T59056 C0RY2G 46233602 IC50 = 43.65 nM T59056 CUV83E 46854605 IC50 = 3450 nM T59056 CIA08B 46854608 IC50 = 974 nM T59056 CWJ3F1 46854758 IC50 = 3830 nM T59056 CKRQ67 46854759 IC50 = 1130 nM T59056 CZ1YJ0 46854760 IC50 = 49500 nM T59056 CIC9S5 49799473 IC50 = 1870 nM T59056 CN6M5D 49820901 IC50 = 1.1 nM T59056 C3Q6AS 49862488 IC50 = 2.5 nM T59056 CM43HV 49862547 IC50 = 5.2 nM T59056 CFDH59 49862548 IC50 = 18.6 nM T59056 CNIA98 49862549 IC50 = 104 nM T59056 CKY2J9 49862550 IC50 = 121 nM T59056 C0N4RT 49862551 IC50 > 1000 nM T59056 CLI23H 49862552 IC50 = 758 nM T59056 CGU86D 49862599 IC50 = 117 nM T59056 CY8WD5 49862600 IC50 = 628 nM T59056 CS4IP9 49862601 IC50 = 9.4 nM T59056 C63XUS 49862602 IC50 = 61.7 nM T59056 C6O7JQ 49862603 IC50 = 11.4 nM T59056 C8G7FR 49862604 IC50 = 7.8 nM T59056 CP5D8Q 49862650 IC50 = 0.9 nM T59056 C6X0JA 49862651 IC50 = 0.8 nM T59056 C7BTK9 49862652 IC50 = 1.3 nM T59056 C79MQZ 49862653 IC50 = 2.4 nM T59056 CL8DR6 49862654 IC50 = 0.3 nM T59056 CH4PA0 51032277 IC50 = 9 nM T59056 CMXR96 51355428 IC50 = 250 nM T59056 C5KTL3 51355429 IC50 = 200 nM T59056 C4UTM8 51355430 IC50 = 101 nM T59056 CH5C9K 51355431 IC50 = 150 nM T59056 CRK2Q9 51355432 IC50 = 125 nM T59056 CF7RG5 51355433 IC50 = 100 nM T59056 C41SUK 51355703 IC50 = 200 nM T59056 CM6T7H 51355704 IC50 = 124 nM T59056 CZDA87 51355705 IC50 = 250 nM T59056 CO1V0Y 51355706 IC50 = 200 nM T59056 C2OCG3 51355707 IC50 = 100 nM T59056 CIR0L7 51356252 IC50 = 2190 nM T59056 CY69GL 52450897 IC50 = 632 nM T59056 C6SIG0 52919010 IC50 = 2.5 nM T59056 CMTX50 52936939 IC50 = 4.3 nM T59056 CC7Q8A 52936940 IC50 = 3.6 nM T59056 CTD3M1 52936941 IC50 = 18 nM T59056 C98MZS 52937039 IC50 = 1.2 nM T59056 CZ72GJ 53316510 IC50 = 372 nM T59056 CR7L6V 53317838 IC50 = 290 nM T59056 CD9JL4 53319024 IC50 = 166 nM T59056 CJBC94 53319146 IC50 > 1000 nM T59056 CYN7S9 53319147 IC50 = 353 nM T59056 C6WXT3 53320325 IC50 = 2226 nM T59056 C20LRW 53320468 IC50 = 77 nM T59056 CU80BY 53320469 IC50 > 1000 nM T59056 C1SH0Q 53321768 IC50 > 1000 nM T59056 CEA3Y9 53321769 IC50 > 1000 nM T59056 C90DZC 53322953 IC50 = 23 nM T59056 CU1V2C 53323093 IC50 = 332 nM T59056 CYU1S5 53323094 IC50 > 1000 nM T59056 CS4A9O 53324450 IC50 = 265 nM T59056 C0B7TL 53325759 IC50 = 1903 nM T59056 CVG4U6 53325760 IC50 = 8 nM T59056 CO68YD 53326854 IC50 = 677 nM T59056 C4NU2F 53475401 IC50 = 2075 nM T59056 C51RVD 56645155 IC50 = 16 nM T59056 CG06MB 56645361 IC50 = 4 nM T59056 CUS9L4 56645362 IC50 = 28 nM T59056 C4N0WL 56645363 IC50 = 1.4 nM T59056 CTO1X9 56645364 IC50 = 2.1 nM T59056 C57NSZ 56645568 IC50 = 0.3 nM T59056 C6PUX9 56645570 IC50 = 4.7 nM T59056 CTW6K2 56645571 IC50 = 0.5 nM T59056 CX05HC 56645572 IC50 = 10.2 nM T59056 CPCW12 56645777 IC50 = 1.2 nM T59056 C32FWC 56645967 IC50 = 0.8 nM T59056 CXYW61 56645969 IC50 = 0.4 nM T59056 C2AP7F 56646158 IC50 = 0.6 nM T59056 CKWB83 56646160 IC50 = 2.2 nM T59056 CH8CP7 57329709 IC50 = 782 nM T59056 CQD5B4 57329785 IC50 = 2832 nM T59056 C8GUF0 57329786 IC50 = 830 nM T59056 CE4YX9 57329787 IC50 = 1157 nM T59056 CRAD59 57329788 IC50 = 1736 nM T59056 CH8FQ9 57329789 IC50 = 2114 nM T59056 C4USR5 57329791 IC50 = 968 nM T59056 C2C5PD 57329792 IC50 = 1243 nM T59056 C3D8CZ 57329793 IC50 = 251 nM T59056 CKH02M 57329866 IC50 = 911 nM T59056 C30NOK 57329940 IC50 = 200 nM T59056 C37KZO 57329941 IC50 = 92 nM T59056 CZH28K 57329942 IC50 = 28 nM T59056 CR6EH0 57329943 IC50 = 220 nM T59056 CWN9V2 57329944 IC50 = 273 nM T59056 CFLA57 57330005 IC50 = 151 nM T59056 C2JR3S 57330006 IC50 = 31 nM T59056 C1EZM8 57330007 IC50 = 110 nM T59056 C5H2LE 57330008 IC50 = 74 nM T59056 C05XKT 57330009 IC50 = 621 nM T59056 C26GFC 57330010 IC50 = 322 nM T59056 CS38WC 57330011 IC50 = 23 nM T59056 C54EUF 57330012 IC50 > 5000 nM T59056 C4MN9B 57330078 IC50 = 4539 nM T59056 C5K3VT 57330079 IC50 = 3111 nM T59056 C3LVG9 57330084 IC50 = 1025 nM T59056 CMNH08 57330085 IC50 = 19 nM T59056 CY58ZD 57330086 IC50 = 33 nM T59056 C7OK1X 57775654 IC50 = 588 nM T59056 CQ0M7J 58215635 IC50 = 3.7 nM T59056 CXH24K 58215717 IC50 = 2 nM T59056 C2AIC8 58215744 IC50 = 5 nM T59056 C78KDY 58215749 IC50 = 4 nM T59056 C9THW1 58215779 IC50 = 90 nM T59056 C96KYA 58215794 IC50 = 11 nM T59056 CB6RN7 58255346 IC50 = 33 nM T59056 CFXY47 58255349 IC50 = 18 nM T59056 C34JIZ 58255359 IC50 = 204 nM T59056 C7ZH6D 58255361 IC50 = 4.2 nM T59056 C2TUJ7 58255382 IC50 = 24 nM T59056 CMBV34 58255389 IC50 = 19 nM T59056 C3DPC0 58255407 IC50 = 104 nM T59056 C9DK1X 58255415 IC50 = 674 nM T59056 CQEW75 58255430 IC50 = 304 nM T59056 CTI0D7 58255435 IC50 = 390 nM T59056 C7L1NK 58255436 IC50 = 29 nM T59056 CRQ70M 58255438 IC50 = 3.8 nM T59056 C72VNQ 58255447 IC50 = 5.8 nM T59056 CLQ65O 58255479 IC50 = 563 nM T59056 CP6RA9 58255482 IC50 = 312 nM T59056 C6DHG3 58255496 IC50 = 308 nM T59056 CAJ17Z 58255506 IC50 = 18 nM T59056 C7AX1R 58255531 IC50 = 88 nM T59056 CJX70M 58255566 IC50 = 85 nM T59056 C64JZC 58255572 IC50 = 851 nM T59056 CW71EO 58255581 IC50 = 268 nM T59056 CYD9N5 58255637 IC50 = 47 nM T59056 COR5V1 58827040 IC50 = 464 nM T59056 C1L8ME 58827183 IC50 = 2 nM T59056 CGZ4S2 58827192 IC50 = 792 nM T59056 CL9G1Q 58827222 IC50 = 390 nM T59056 C7FK9X 59534652 IC50 = 380 nM T59056 CCX31E 59578413 IC50 = 22 nM T59056 CB7N8A 60195126 IC50 = 100 nM T59056 CX4N0I 62707515 IC50 = 19 nM T59056 CH3QU4 62918897 IC50 > 1000 nM T59056 CE6L7O 65040275 IC50 = 1768 nM T59056 C0G3LA 66559847 IC50 = 19 nM T59056 C4RSI6 66559935 IC50 = 1703 nM T59056 CDX7I8 66559936 IC50 = 759 nM T59056 CF9EQ5 66559939 IC50 = 12 nM T59056 CQN6D3 66559940 IC50 = 1167 nM T59056 CN4H8G 66559941 IC50 = 1097 nM T59056 CTP6Q4 66559942 IC50 = 208 nM T59056 C9EGW2 66575742 IC50 = 57.2 nM T59056 CMXA10 66575743 IC50 = 4.2 nM T59056 CKWB91 66575744 IC50 = 2.2 nM T59056 C7I3MW 66575745 IC50 = 62.5 nM T59056 CPN17S 66575746 IC50 = 131.4 nM T59056 CG0ZA7 66575747 IC50 = 172.2 nM T59056 C6HF0U 66575748 IC50 = 244 nM T59056 CEW4O6 66575816 IC50 = 41 nM T59056 CDI93T 66575817 IC50 = 7.1 nM T59056 C6B7PN 66576767 IC50 = 5 nM T59056 CYHS25 66576769 IC50 = 40 nM T59056 CBP6I7 66576773 IC50 = 58 nM T59056 CM6U5S 66576848 IC50 = 22 nM T59056 CNB21T 66576849 IC50 = 17 nM T59056 C2PFB6 66576850 IC50 = 32 nM T59056 CDU8R7 66576852 IC50 = 48 nM T59056 C4NYB0 66576930 IC50 = 20.3 nM T59056 C3LP5H 66576931 IC50 = 28.3 nM T59056 CE03WG 66576932 IC50 = 87.6 nM T59056 CVZ4E0 66692998 IC50 > 1000 nM T59056 C1RLT0 67199421 IC50 = 366 nM T59056 CC34QF 67509960 IC50 = 25 nM T59056 CQL7H6 67510362 IC50 = 5159 nM T59056 CN9VU2 67510431 IC50 > 1000 nM T59056 C40FEA 67511528 IC50 = 929 nM T59056 C2MH1G 67515607 IC50 = 3265 nM T59056 CC4A7Z 67515696 IC50 = 528 nM T59056 CE27NZ 67515801 IC50 > 1000 nM T59056 CZCW84 67515869 IC50 = 851 nM T59056 CKJN74 67515874 IC50 > 1000 nM T59056 CW20PM 67516106 IC50 = 3955 nM T59056 C14VNF 67516160 IC50 > 1000 nM T59056 CM7Z1T 67516370 IC50 = 914 nM T59056 CK1LB2 67516475 IC50 > 1000 nM T59056 C5VM6T 67516855 IC50 = 487 nM T59056 CQ0NP7 68053462 IC50 > 1000 nM T59056 CV72CY 68053552 IC50 = 24 nM T59056 CI0PN4 68053567 IC50 = 0.15 nM T59056 CVF40X 68053622 IC50 = 254 nM T59056 CG0T8B 68053623 IC50 = 35 nM T59056 CU76KO 68053624 IC50 = 561 nM T59056 CYZK18 68053631 IC50 = 219 nM T59056 CSI12Z 68053632 IC50 = 107 nM T59056 C0N3IK 68053729 IC50 = 0.2 nM T59056 C19JSA 68053730 IC50 = 0.4 nM T59056 C5N2MQ 68053837 IC50 = 12 nM T59056 CCJT39 68053838 IC50 = 138 nM T59056 CF32HJ 70680985 IC50 > 1000 nM T59056 CPB63L 70680997 IC50 = 416 nM T59056 CE78SM 70683110 IC50 = 576 nM T59056 CM6LN8 70683111 IC50 > 1000 nM T59056 C9E4ZQ 70685192 IC50 = 281 nM T59056 CW5F3G 70691516 IC50 > 1000 nM T59056 C1VMF2 70977969 IC50 = 89.7 nM T59056 CF9O7Z 71114804 IC50 = 5000 nM T59056 CW0JS9 71114814 IC50 = 7000 nM T59056 C70TUP 71455138 IC50 = 178 nM T59056 CFG4L5 71456934 IC50 = 22 nM T59056 CI16NC 71520311 IC50 = 41 nM T59056 CE9A6B 71520312 IC50 = 1580 nM T59056 C03VKJ 71520313 IC50 > 5000 nM T59056 C5J7DI 71520314 IC50 = 74 nM T59056 CE0N5C 71520315 IC50 = 468 nM T59056 C4Z6YP 71520316 IC50 = 96 nM T59056 CC8Z6L 71520431 IC50 = 37 nM T59056 C1DK9P 71520432 IC50 = 74 nM T59056 C9NOQ1 71521632 IC50 = 132 nM T59056 C0OTA2 71521716 IC50 > 5000 nM T59056 CVLE07 71521717 IC50 > 5000 nM T59056 CJKX84 71521718 IC50 > 5000 nM T59056 CZ5P9U 71521719 IC50 = 587 nM T59056 C1YCB0 71521720 IC50 = 750 nM T59056 CE57PM 71521721 IC50 = 1290 nM T59056 C0O2SA 71521798 IC50 = 128 nM T59056 CMEC10 71521799 IC50 = 139 nM T59056 CR9O5T 71521800 IC50 = 46 nM T59056 C0JBI3 71521801 IC50 = 88 nM T59056 CE7Z4I 71521802 IC50 = 56 nM T59056 CW2AG4 71521803 IC50 = 51 nM T59056 C6ID7K 71521804 IC50 = 32 nM T59056 CO5BE7 71535395 IC50 = 3.3 nM T59056 CCF8Z7 71535398 IC50 = 4 nM T59056 CC16AO 71535399 IC50 = 10 nM T59056 CPZ5S8 71535400 IC50 = 0.6 nM T59056 CI4W5N 71535682 IC50 = 33 nM T59056 CCRS95 71535683 IC50 = 25 nM T59056 C58SMB 71574941 IC50 = 3 nM T59056 CC09FQ 71574942 IC50 = 23.5 nM T59056 CA2T5L 71574943 IC50 = 103.9 nM T59056 C9MFZ7 71574944 IC50 = 41.1 nM T59056 CW73OE 71574945 IC50 = 14.8 nM T59056 C70NHJ 71574946 IC50 = 19.1 nM T59056 CLH83S 71574947 IC50 = 25.2 nM T59056 CF71AB 71575030 IC50 = 15.3 nM T59056 CCG1S5 71575031 IC50 = 24.1 nM T59056 CH9WE7 71575032 IC50 = 99.7 nM T59056 CO4ZQ7 71575033 IC50 = 235.3 nM T59056 CT86GV 71575034 IC50 = 676.5 nM T59056 CKPV51 71621803 IC50 > 100000 nM T59056 CG09JH 71716351 IC50 = 1736 nM T59056 C56LUJ 71716957 IC50 = 5 nM T59056 CJE01S 71745100 IC50 = 19.5 nM T59056 CZMQ02 71811360 IC50 = 42 nM T59056 CH8M5Y 71811363 IC50 = 25 nM T59056 C1WT8V 71811365 IC50 = 21 nM T59056 CIK35Q 71811651 IC50 = 47 nM T59056 C1B5VY 71811696 IC50 = 27 nM T59056 C3VK0H 71811699 IC50 = 14 nM T59056 CX0WV5 71817943 IC50 = 26 nM T59056 CN1LU6 71817944 IC50 = 17 nM T59056 CGV4U3 71817945 IC50 = 30 nM T59056 CJ4L5G 71818086 IC50 = 28 nM T59056 COXA51 71818087 IC50 = 25 nM T59056 CP1A3M 71818088 IC50 = 38 nM T59056 CPJ42T 71818089 IC50 = 33 nM T59056 CAP03I 71818090 IC50 = 24 nM T59056 CO23PK 71818091 IC50 = 15 nM T59056 CL4X6A 71818092 IC50 = 13 nM T59056 CL8GK5 71818093 IC50 = 27 nM T59056 C4ZVG0 71818094 IC50 = 54 nM T59056 CH2GR0 71818232 IC50 = 66 nM T59056 C0VGQ9 71818233 IC50 = 72 nM T59056 C5QRF2 71818234 IC50 = 22 nM T59056 C7NV1F 72724763 IC50 = 87 nM T59056 C4AEX3 73347616 IC50 = 1115 nM T59056 CFD46C 73347617 IC50 = 25 nM T59056 C26LJW 73347618 IC50 = 1880 nM T59056 CIHF35 73350707 IC50 = 836 nM T59056 CT26EZ 73355186 IC50 > 5000 nM T59056 C0NXU4 73355187 IC50 = 302 nM T59056 CML29U 73355188 IC50 = 2924 nM T59056 CC5TO4 73356735 IC50 = 419 nM T59056 CWZ3A1 73356736 IC50 = 0.5 nM T59056 C9CY3K 73442767 IC50 = 0.6 nM T59056 CU6IQ9 73603293 IC50 = 228 nM T59056 C6MQ8L 73603294 IC50 > 5000 nM T59056 CR81XZ 73603295 IC50 = 1285 nM T59056 CJS6Y2 73603296 IC50 = 2833 nM T59056 C1GR7W 73603297 IC50 = 1433 nM T59056 CM4L6N 73603298 IC50 > 5000 nM T59056 CAIB62 73603299 IC50 = 3070 nM T59056 C7G6KZ 73603343 IC50 = 0.7 nM T59056 CDX9R1 73603344 IC50 = 2.8 nM T59056 C7KV2S 73603345 IC50 = 152 nM T59056 CM10ZX 73603346 IC50 = 30 nM T59056 CJSY07 73603348 IC50 = 23 nM T59056 CS03UP 73603349 IC50 = 61 nM T59056 C56LYP 73603350 IC50 = 426 nM T59056 C9RKH0 73603387 IC50 = 16 nM T59056 CG86BD 73603388 IC50 = 36 nM T59056 C2R3ZB 73603389 IC50 = 55 nM T59056 C5ARE7 73603390 IC50 = 3 nM T59056 CTMF86 73603391 IC50 = 2.2 nM T59056 C5RG4C 75593332 IC50 = 0.9 nM T59056 CMN51L 76286753 IC50 = 217 nM T59056 C06HYT 76286902 IC50 = 44 nM T59056 CS80JY 76310075 IC50 = 17 nM T59056 CL13PY 76310076 IC50 = 140 nM T59056 CRQW60 76310077 IC50 = 10 nM T59056 C7C3EM 76313777 IC50 = 16 nM T59056 CM26XC 76313778 IC50 = 520 nM T59056 CE65PA 76313779 IC50 = 56 nM T59056 CPU3T6 76317295 IC50 = 3.2 nM T59056 C0GE4M 76317296 IC50 = 37 nM T59056 CXK20H 76320999 IC50 = 441 nM T59056 CZ2U9K 76321000 IC50 = 8 nM T59056 CB74PI 76324668 IC50 = 2 nM T59056 C1O4CX 76324671 IC50 = 351 nM T59056 C30WIM 76324672 IC50 = 5 nM T59056 CQM6E9 76328229 IC50 = 3 nM T59056 CBC64P 76328230 IC50 = 13 nM T59056 C4UO5H 76331904 IC50 = 1.5 nM T59056 CW7C5H 76331905 IC50 = 5 nM T59056 C32BDK 76335487 IC50 = 2 nM T59056 CP10SN 76335488 IC50 = 0.4 nM T59056 C2ASY0 86730379 IC50 = 52 nM T59056 CA4QV9 86730380 IC50 = 1.2 nM T59056 C24ZMT 86730381 IC50 = 1.2 nM T59056 C9W6RO 86730382 IC50 = 23 nM T59056 C3UMP9 89471867 IC50 = 2.5 nM T59056 CW8TF6 89471869 IC50 = 6.6 nM T59056 CL30TR 89471870 IC50 = 7.3 nM T59056 CJ0H5V 89471872 IC50 = 23 nM T59056 C3BUS8 89471889 IC50 = 7.9 nM T59056 CI7HY8 89471890 IC50 = 6.6 nM T59056 CF2AY7 89471891 IC50 = 160 nM T59056 CQF07X 89471892 IC50 = 13 nM T59056 CA3G9X 89600687 IC50 = 2.8 nM T59056 CAC8M9 89846231 IC50 = 28 nM T59056 C16AXO 89846366 IC50 = 123 nM T59056 CEK2I7 89846957 IC50 = 942 nM T59056 C4MJ6O 89846958 IC50 = 9 nM T59056 C62KFZ 89961587 IC50 = 486 nM T59056 C8XS2I 89961629 IC50 = 19 nM T59056 C75PMO 89961672 IC50 = 506 nM T59056 CX0M7B 89961716 IC50 = 103 nM T59056 C3JN5I 89961721 IC50 = 423 nM T59056 CSJT14 89961765 IC50 = 526 nM T59056 CR5D6Y 89961785 IC50 = 335 nM T59056 C7TI3V 89961787 IC50 = 2400 nM T59056 C2QP7I 89961848 IC50 = 487 nM T59056 C81FEN 89961879 IC50 = 300 nM T59056 CI6P0R 89961978 IC50 = 283 nM T59056 C89TEU 89968659 IC50 = 42.5 nM T59056 C7BC5N 89968688 IC50 = 558 nM T59056 C3XIF5 90252771 IC50 = 0.2 nM T59056 CGZ2S1 90252806 IC50 = 27 nM T59056 C4F9VB 90252809 IC50 = 25 nM T59056 CE2TM0 90252810 IC50 = 528 nM T59056 CGVL78 90252811 IC50 = 2300 nM T59056 C0S3HV 90252812 IC50 = 97.9 nM T59056 C4M8TO 90252814 IC50 = 507 nM T59056 CM0T2X 90252815 IC50 = 1156 nM T59056 CY5IC7 90252834 IC50 = 2.2 nM T59056 CF05JI 90252835 IC50 = 84.9 nM T59056 C72ICB 90252839 IC50 = 456 nM T59056 C84NVA 90252850 IC50 = 14 nM T59056 CBY46O 90252851 IC50 = 77 nM T59056 CNVA50 90252852 IC50 = 32.9 nM T59056 C0Z2TI 90252864 IC50 = 2 nM T59056 CV30CD 90252953 IC50 = 15 nM T59056 C3MV7S 90252954 IC50 = 88 nM T59056 CD5ST8 90252956 IC50 = 760 nM T59056 C3JH4P 90252957 IC50 = 300 nM T59056 CCU4F7 90252958 IC50 = 78.5 nM T59056 C82YUB 90644545 IC50 = 14 nM T59056 CVFA18 90644546 IC50 = 77 nM T59056 CR50EN 90644547 IC50 = 1.7 nM T59056 C46ZNM 90644548 IC50 = 13 nM T59056 CS6N1P 90644549 IC50 > 5000 nM T59056 CB5HI4 90644550 IC50 = 5 nM T59056 CLB2E7 91827654 IC50 = 64 nM T59056 C5GV1L 101882447 IC50 = 5 nM T59056 CMH51N 118496543 IC50 = 33.5 nM T59056 C3ZPQ1 118496545 IC50 = 7.58 nM T59056 CJ9Z0S 118496546 IC50 = 1.3 nM T59056 C7UN3R 118496547 IC50 = 10.9 nM T59056 C1RE7O 118496557 IC50 = 22 nM T59056 C3WKQ5 118707346 IC50 = 1.4 nM T59056 CP92XR 118707348 IC50 = 21 nM T59056 CNSW38 118707349 IC50 = 5 nM T59056 CLS25A 118714825 IC50 = 5 nM T59056 CT0FH7 118714826 IC50 = 5 nM T59056 CD8T1P 118714827 IC50 = 5 nM T59056 C85BVO 118714828 IC50 = 5 nM T59056 CYFP62 118714829 IC50 = 5 nM T59056 CE3ZF1 118714830 IC50 = 5 nM T59056 C5HKE1 118714831 IC50 = 5 nM T59056 C7BD3X 118714832 IC50 = 5 nM T59056 C9BM7X 118714833 IC50 = 5 nM T59056 CML4K7 118714834 IC50 = 5 nM T59056 CE5L8U 118714835 IC50 = 5 nM T59056 CD8YA9 118714836 IC50 = 5 nM T59056 CRNL64 118714837 IC50 = 5 nM T59056 C4F6AY 118714838 IC50 = 5 nM T59056 CZ9L5S 118714839 IC50 = 5 nM T59056 CU3XP2 118714840 IC50 = 5 nM T59056 C0BRP1 118714841 IC50 = 5 nM T59056 C6M5VU 118714842 IC50 = 5 nM T59056 CQ5KI0 118714843 IC50 = 5 nM T59056 C32MDK 118714844 IC50 = 5 nM T59056 C15PAW 118714845 IC50 = 5 nM T59056 CPH51S 118714846 IC50 = 5 nM T59056 C1L4YZ 118714847 IC50 = 5 nM T59056 CLM64U 118714848 IC50 = 5 nM T59056 C5UD3K 118714849 IC50 = 5 nM T59056 CNW8E3 118714850 IC50 = 5 nM T59056 CMXG03 118714851 IC50 = 5 nM T59056 CTWO23 118714852 IC50 = 5 nM T59056 CAW36P 118714853 IC50 = 5 nM T59056 C4Y2UF 118714854 IC50 = 5 nM T59056 CJK08Q 118714855 IC50 = 5 nM T59056 CP4O0C 118720463 IC50 = 33 nM T59056 CV4IC9 118720464 IC50 = 48 nM T59056 CKG28R 118720465 IC50 = 27 nM T59056 CGXD81 118720466 IC50 = 64 nM T59056 CF1W7I 118720467 IC50 = 22 nM T59056 COZU39 118720468 IC50 = 60 nM T59056 CWG6L8 118720469 IC50 = 22 nM T59056 C2HV3Y 118720470 IC50 = 33 nM T59056 CX56BZ 118720471 IC50 = 39 nM T59056 CO8H3J 118720472 IC50 = 32 nM T59056 C7WEQ3 118720473 IC50 = 14 nM T59056 CG8PB5 118720474 IC50 = 56 nM T59056 CN2U6B 118720475 IC50 = 25 nM T59056 CU7FW1 118720476 IC50 = 43 nM T59056 CCJ17Z 118720477 IC50 = 53 nM T59056 CB4DS9 118720479 IC50 = 46 nM T59056 CC9V6K 118720480 IC50 = 33 nM T59056 CP7X1B 118720481 IC50 = 33 nM T59056 CPT58L 118720482 IC50 = 47 nM T59056 C3E7TA 118720483 IC50 = 53 nM T59056 CS01NU 118720484 IC50 = 192 nM T59056 CAW5K3 118723935 IC50 = 127 nM T59056 CK8UL1 118723936 IC50 = 86 nM T59056 CIW7O0 118723937 IC50 = 77 nM T59056 C42CEZ 118723938 IC50 = 82 nM T59056 CJQ63E 118723939 IC50 = 899 nM T59056 CCXN71 118723940 IC50 = 82 nM T59056 CS78BD 118723941 IC50 = 147 nM T59056 C9W3QX 118723942 IC50 > 500 nM T59056 COJ2K8 118723943 IC50 = 497 nM T59056 CZ23UL 118723944 IC50 = 192 nM T59056 CIWU64 118723945 IC50 = 222 nM T59056 CZI6A0 118723946 IC50 = 669 nM T59056 COB46M 118723947 IC50 = 1397 nM T59056 CYM08W 118726850 IC50 = 228 nM T59056 CR32JU 118726851 IC50 = 2.2 nM T59056 C2OAI6 118726852 IC50 = 193 nM T59056 CDHI10 118733086 IC50 = 979.3 nM T59056 C18PWB 118733087 IC50 = 541.7 nM T59056 C8WJ2Y 118733088 IC50 > 10000 nM T59056 C31ZXP 118733089 IC50 > 10000 nM T59056 CHR84E 118733090 IC50 > 10000 nM T59056 CAQ72M 118733091 IC50 > 10000 nM T59056 CIV1Z5 118733092 IC50 = 4354.4 nM T59056 CU3Y9W 118733093 IC50 = 707.7 nM T59056 CF49NU 118733094 IC50 > 10000 nM T59056 CK73VU 118733095 IC50 > 10000 nM T59056 CR1WU5 118733096 IC50 = 1177.9 nM T59056 C1V7WI 118735163 IC50 = 643 nM T59056 C6YG9R 118735164 IC50 = 756 nM T59056 C5C4FZ 118735165 IC50 = 260 nM T59056 C1ZLM6 118735166 IC50 = 17 nM T59056 CQXM57 118735167 IC50 = 53 nM T59056 C0RYM4 118735168 IC50 = 15 nM T59056 C0DCB9 118735169 IC50 = 87 nM T59056 CG4QF3 118735170 IC50 = 7 nM T59056 CD3IY5 118735171 IC50 = 18 nM T59056 C0JZ2Y 118735172 IC50 = 447 nM T59056 C2WS7A 118735173 IC50 = 714 nM T59056 CYEA24 118735174 IC50 = 84 nM T59056 CZ9X4J 118735175 IC50 = 74 nM T59056 CG14RD 118735176 IC50 = 230 nM T59056 CQ3KR4 118735177 IC50 = 70 nM T59056 C1Z9FX 118735178 IC50 = 945 nM T59056 C2VJU4 118735179 IC50 = 24 nM T59056 CXWH51 118735180 IC50 = 63 nM T59056 C3YUS9 118735181 IC50 = 23 nM T59056 CEH97S 118735182 IC50 = 299 nM T59056 C03HKR 118735183 IC50 = 816 nM T59056 CC38HG 118735184 IC50 = 1453 nM T59056 C8QIC4 118735185 IC50 = 2441 nM T59056 CZET62 118735186 IC50 = 246 nM T59056 CZ8U2C 118735187 IC50 = 16 nM T59056 CUAE09 121004872 IC50 = 49 nM T59056 C1OT4E 121458684 IC50 = 22.3 nM T59056 C9ETN3 121458685 IC50 = 8.1 nM T59056 C4V2HU 121458987 IC50 = 1 nM T59056 CPGD72 121458994 IC50 = 0.6 nM T59056 CXW13O 122179553 IC50 > 5000 nM T59056 C3E0VM 122179554 IC50 > 5000 nM T59056 CJVX13 122179555 IC50 = 607 nM T59056 CWN9K7 122179556 IC50 > 10000 nM T59056 CV2PQ1 122191831 IC50 > 8333 nM T59056 C2AHB5 122191832 IC50 > 8333 nM T59056 CFZH01 122191833 IC50 > 8333 nM T59056 C1XKA8 122191834 IC50 = 109 nM T59056 CG4S8F 122191835 IC50 = 461 nM T59056 C37NLK 122191836 IC50 = 476 nM T59056 CVT7A2 127027254 IC50 = 213.8 nM T59056 C5QNG6 127027265 IC50 > 10000 nM T59056 CIZO64 127027266 IC50 > 10000 nM T59056 C9RXH3 127027267 IC50 > 10000 nM T59056 CEM84R 127027569 IC50 = 2268.4 nM T59056 CT83ZE 127027570 IC50 = 619.8 nM T59056 CHZ54G 127027571 IC50 = 121.2 nM T59056 C2ZFR8 127027572 IC50 = 1066.1 nM T59056 CV1BD6 127027573 IC50 = 94.9 nM T59056 C0E6DW 127027574 IC50 > 10000 nM T59056 C2MFJ8 127027575 IC50 > 10000 nM T59056 CM8T9G 127028498 IC50 = 3270.6 nM T59056 CQO36B 127028499 IC50 = 317.3 nM T59056 C1M7GD 127028500 IC50 = 1235.3 nM T59056 CN42BR 127028817 IC50 = 643.2 nM T59056 C3IMJ8 127028818 IC50 = 521.5 nM T59056 CPEM69 127028819 IC50 = 767.9 nM T59056 C70XOB 127030295 IC50 > 5000 nM T59056 CZ7L4J 127031191 IC50 > 10000 nM T59056 C49IME 127031799 IC50 = 953.6 nM T59056 CHS8L7 131982520 IC50 = 12 nM T59056 CG9UJ7 131982526 IC50 > 1000 nM T59056 C95PYQ 131982530 IC50 = 3.7 nM T59056 C5IWD9 131982539 IC50 = 29 nM T59056 CSIP72 131982576 IC50 = 3.2 nM T59056 CS8C7T 131982729 IC50 = 4.7 nM T59056 CHDP80 131982862 IC50 = 14 nM T59056 C1BNU6 131982871 IC50 = 71 nM T59056 C6CB0I 132585204 IC50 = 27 nM T59056 C7SM9W 134129925 IC50 = 13 nM T59056 CB3EL1 134134056 IC50 = 42 nM T59056 CB79AO 134134186 IC50 > 10000 nM T59056 CPZX32 134135994 IC50 = 448 nM T59056 CS2P0E 134136577 IC50 = 73 nM T59056 CH3V9Q 134139925 IC50 = 6.6 nM T59056 CFUE13 134141128 IC50 = 554 nM T59056 COUK40 134141967 IC50 = 228 nM T59056 CX3Y9D 134142597 IC50 = 106 nM T59056 CQF59S 134143092 IC50 = 704 nM T59056 C1HG8V 134144349 IC50 = 34 nM T59056 CFC8O6 134145376 IC50 = 5.8 nM T59056 C31WNO 134145695 IC50 = 1134 nM T59056 C7JEU2 134148873 IC50 = 4.7 nM T59056 C2JOB5 134152002 IC50 = 32 nM T59056 CTXL17 134153274 IC50 = 1031 nM T59056 C3OLF2 134153424 IC50 > 8000 nM T59056 C12LPH 134153935 IC50 = 13 nM T59056 C8ROI0 134153997 IC50 = 26 nM T59056 CDV8M5 134155385 IC50 = 98 nM T59056 C74ONC 134156861 IC50 = 94 nM T59056 CKL9N7 135185757 IC50 = 29 nM T59056 C8HTS7 135185761 IC50 = 172 nM T59056 C1D4CS 135185764 IC50 = 40 nM T59056 CMQC50 135185766 IC50 = 3 nM T59056 CIS5H8 135185771 IC50 = 17 nM T59056 CF0EC1 135185786 IC50 = 18 nM T59056 C8GB5V 135185787 IC50 = 9 nM T59056 CH30EN 135185789 IC50 = 8 nM T59056 CMR5C9 135185792 IC50 = 29 nM T59056 CX97YM 135185793 IC50 = 5 nM T59056 CS5FX2 135185796 IC50 = 22 nM T59056 CV9RM5 135185801 IC50 = 13 nM T59056 C8MF2Z 135185815 IC50 < 2 nM T59056 CX57GP 135185833 IC50 = 24 nM T59056 CSZA19 135185836 IC50 = 50 nM T59056 C6G1CH 135185858 IC50 = 25 nM T59056 C9LU0C 135185886 IC50 = 16 nM T59056 CZ1JS3 135186252 IC50 = 330 nM T59056 CWU63C 136008115 IC50 = 237 nM T59056 CZ2YW4 136074307 IC50 = 2.2 nM T59056 CM97FH 137631528 IC50 = 152 nM T59056 C9LY0O 137631806 IC50 = 6 nM T59056 CB35YI 137632879 IC50 = 109 nM T59056 CH05YR 137633095 IC50 = 173 nM T59056 COG72W 137633343 IC50 = 30 nM T59056 C3QE1V 137633417 IC50 = 27 nM T59056 CVM54L 137634483 IC50 = 32 nM T59056 C14ALD 137635413 IC50 = 300 nM T59056 CL1SQ6 137636747 IC50 = 14 nM T59056 CV2S5Q 137637282 IC50 = 8 nM T59056 CUIX95 137637496 IC50 = 7.77 nM T59056 C14LXC 137638585 IC50 = 5 nM T59056 C1D0WG 137638612 IC50 = 24 nM T59056 CF1D5C 137639549 IC50 = 2 nM T59056 C8V7CD 137639692 IC50 = 2 nM T59056 C1SH2M 137639834 IC50 = 0.3 nM T59056 CZA2S8 137639890 IC50 = 120 nM T59056 C0N4PJ 137640302 IC50 = 48 nM T59056 COEV02 137642385 IC50 = 3 nM T59056 CH35RE 137642529 IC50 = 0.4 nM T59056 CP1EJ0 137642735 IC50 = 90 nM T59056 C29FMO 137642787 IC50 = 586 nM T59056 COGQ01 137644314 IC50 = 97 nM T59056 CA73KP 137644560 IC50 = 520 nM T59056 C5DH8X 137645356 IC50 = 83 nM T59056 C4UP3J 137647900 IC50 = 4 nM T59056 CI31EQ 137649226 IC50 = 507 nM T59056 CRF41D 137649685 IC50 = 144 nM T59056 CS5BW7 137650545 IC50 = 28 nM T59056 CF71RE 137650772 IC50 = 657 nM T59056 CQ54YG 137651298 IC50 = 82 nM T59056 C4CL2W 137651728 IC50 = 15 nM T59056 CK7QJ4 137651744 IC50 = 17 nM T59056 C4A9QW 137652329 IC50 = 300 nM T59056 CI5D2P 137652926 IC50 = 30 nM T59056 CIH34U 137653629 IC50 = 31 nM T59056 CV9I5G 137653991 IC50 = 5 nM T59056 C28VRO 137654883 IC50 = 8 nM T59056 CEV94S 137655303 IC50 = 1304 nM T59056 CY5IK7 137655531 IC50 = 16 nM T59056 CUL37V 137655879 IC50 = 8 nM T59056 CN2CQ1 137656473 IC50 = 459 nM T59056 C53NVI 137657989 IC50 = 24 nM T59056 CNI0C1 137658011 IC50 = 182 nM T59056 C32WHO 137658276 IC50 = 75 nM T59056 C0G2UI 137658690 IC50 = 215 nM T59056 CLNU74 137659288 IC50 = 174 nM T59056 CQNA81 137659369 IC50 = 192 nM T59056 CA5LI1 137659926 IC50 = 116 nM T59056 C7YI9N 137660712 IC50 = 3 nM T59056 CFU1Z3 145960404 IC50 = 2.2 nM T59056 C1IU5W 145960520 IC50 = 9.2 nM T59056 CI5AU7 145960748 IC50 > 1000 nM T59056 CQFH90 145960862 IC50 = 6.7 nM T59056 CNIB73 145960902 IC50 = 5.4 nM T59056 C0KNY4 145961099 IC50 = 2.3 nM T59056 CGI39P 145961215 IC50 = 26 nM T59056 CW84OQ 145961259 IC50 = 290 nM T59056 C92JOV 145961758 IC50 = 150 nM T59056 CR6JH8 145961916 IC50 = 34 nM T59056 CS4EO5 145962296 IC50 = 4.2 nM T59056 C1O0NQ 145962517 IC50 = 13 nM T59056 C6VO0A 145962577 IC50 = 2.2 nM T59056 CY20CQ 145962664 IC50 > 1000 nM T59056 C6F7UE 145962949 IC50 = 2.5 nM T59056 C5O4RQ 145963242 IC50 = 280 nM T59056 CGA01F 145963470 IC50 = 4 nM T59056 CH0TM7 145963574 IC50 = 72 nM T59056 C0TZR1 145964456 IC50 = 135.1 nM T59056 CRJM82 145965429 IC50 = 95.3 nM T59056 CN7B1I 145968025 IC50 = 82 nM T59056 C82JTH 145971322 IC50 = 44.4 nM T59056 C5R6SH 145973507 IC50 = 20.3 nM T59056 C41LQE 145976039 IC50 = 22.3 nM T59056 C01TYI 145976345 IC50 = 45.4 nM T59056 CG23BW 145977901 IC50 = 26.2 nM T59056 C65ZFY 145978611 IC50 = 16.6 nM T59056 CH6DJ3 155527950 IC50 = 62 nM T59056 C80XNT 155530085 IC50 = 782 nM T59056 C5XB1F 155530577 IC50 > 10000 nM T59056 C6DXN8 155559405 IC50 = 412 nM T59056 C4UQS2 155564575 IC50 = 541 nM T59056 CXM62E 155566406 IC50 = 1064 nM T59056 D00BVP 11847320 IC50 = 11 nM T59056 D00DSE 49864196 IC50 = 515 nM T59056 D00PXF 44206698 IC50 = 5.495 nM T59056 D01JZO 2779191 IC50 = 46 nM T59056 D01REI 46901610 IC50 = 948 nM T59056 D01SUE 6539759 IC50 = 11 nM T59056 D01SZX 46867545 IC50 = 114.3 nM T59056 D02ALK 11514074 IC50 = 23 nM T59056 D02BWQ 6539818 IC50 = 41 nM T59056 D02BXS 46901445 IC50 = 367 nM T59056 D02CSU 6539786 IC50 = 18 nM T59056 D02GFK 25034431 IC50 = 13 nM T59056 D02JUJ 25034344 IC50 = 94 nM T59056 D02LWB 6540046 IC50 = 13 nM T59056 D02NAG 6539765 IC50 = 26 nM T59056 D02PSL 45103913 IC50 = 5.2 nM T59056 D02UZI 6540056 IC50 = 735 nM T59056 D02XHH 6540043 IC50 = 10.3 nM T59056 D02XTS 6539811 IC50 = 9 nM T59056 D02ZQM 25180104 IC50 = 44 nM T59056 D03CWL 14535954 IC50 = 193 nM T59056 D03EXD 49864181 IC50 = 341 nM T59056 D03KLN 11413434 IC50 = 19 nM T59056 D03MKT 6539788 IC50 = 15 nM T59056 D03TRM 6540032 IC50 = 41 nM T59056 D03VRC 2989557 IC50 = 479 nM T59056 D03YHZ 25147692 IC50 = 0.2 nM T59056 D04CFP 46901927 IC50 = 231 nM T59056 D04CLL 6539775 IC50 = 108 nM T59056 D04ELJ 6539766 IC50 = 73 nM T59056 D04IBH 11616637 IC50 = 33 nM T59056 D04IJE 256445 IC50 = 5 nM T59056 D04ISG 11680597 IC50 = 29 nM T59056 D04PKP 23644953 IC50 = 14 nM T59056 D04QPK 6539783 IC50 = 21 nM T59056 D04WJN 10588478 IC50 = 344.1 nM T59056 D05FFY 14231155 IC50 = 12 nM T59056 D05IXU 25130517 IC50 = 154 nM T59056 D05MQE 6539785 IC50 = 31 nM T59056 D05QPR 12229388 IC50 = 330 nM T59056 D05YNW 6539790 IC50 = 8 nM T59056 D06CWR 24754344 IC50 = 0.6 nM T59056 D06HFV 6539805 IC50 = 6 nM T59056 D06JYY 25130848 IC50 = 7.8 nM T59056 D06NFC 45103808 IC50 = 10.96 nM T59056 D06RSD 45103911 IC50 = 407.38 nM T59056 D07CTI 10853186 IC50 = 31.1 nM T59056 D07DQJ 45103810 IC50 = 5.1 nM T59056 D07EJK 10632289 IC50 = 61.66 nM T59056 D07IQG 10473365 IC50 = 8.5 nM T59056 D07JCO 12354256 IC50 = 604 nM T59056 D07JMO 10220337 IC50 = 363.08 nM T59056 D07NAH 21772021 IC50 = 296 nM T59056 D07PYC 6539760 IC50 = 92 nM T59056 D07SOM 11847316 IC50 = 28 nM T59056 D07VGT 46901929 IC50 = 1130 nM T59056 D07WLT 25180108 IC50 = 7.8 nM T59056 D07ZCD 6539804 IC50 = 8 nM T59056 D07ZYL 6539797 IC50 = 55 nM T59056 D08AZK 6539767 IC50 = 37 nM T59056 D08EZA 11847317 IC50 = 95 nM T59056 D08FAB 11845485 IC50 = 28 nM T59056 D08HHA 19902087 IC50 = 812.83 nM T59056 D08HPU 6540052 IC50 = 5 nM T59056 D08IDC 24827305 IC50 = 4.2 nM T59056 D08ORG 10198247 IC50 = 28.84 nM T59056 D08PNF 6539770 IC50 = 26 nM T59056 D08WHC 10397593 IC50 = 1174.9 nM T59056 D08YGW 10444038 IC50 = 11 nM T59056 D08ZTZ 11529133 IC50 = 13 nM T59056 D09CPC 13728862 IC50 = 28 nM T59056 D09HEA 1236449 IC50 = 371.54 nM T59056 D09HGK 6539796 IC50 = 59 nM T59056 D09HOE 6539789 IC50 = 29 nM T59056 D09QDY 6540033 IC50 = 11 nM T59056 D09VPA 6539794 IC50 = 24 nM T59056 D09VQZ 46901616 IC50 = 273 nM T59056 D09YXV 6539769 IC50 = 34 nM T59056 D09ZHX 11847318 IC50 = 25 nM T59056 D0AK9S 22466877 IC50 = 6.166 nM T59056 D0AW7Q 46867544 IC50 = 1140.4 nM T59056 D0B2UM 25034430 IC50 = 0.8 nM T59056 D0C6US 6540055 IC50 = 2834 nM T59056 D0C7YL 6481821 IC50 = 600 nM T59056 D0C8EO 6539806 IC50 = 17 nM T59056 D0D7YL 11586681 IC50 = 10 nM T59056 D0D8GU 6539803 IC50 = 4 nM T59056 D0D8KN 45103805 IC50 = 286 nM T59056 D0D8YE 6540048 IC50 = 4 nM T59056 D0D9FR 6539795 IC50 = 56 nM T59056 D0E0ZS 46901613 IC50 = 567 nM T59056 D0E8DX 25180300 IC50 = 3.1 nM T59056 D0E9WX 6540042 IC50 = 92.8 nM T59056 D0F5AC 46867542 IC50 = 43.7 nM T59056 D0F5YU 6539793 IC50 = 36 nM T59056 D0G6QL 23644748 IC50 = 38.5 nM T59056 D0G9WP 18407230 IC50 = 4.4 nM T59056 D0HL9S 1265319 IC50 = 1000 nM T59056 D0I1YH 46901446 IC50 = 261 nM T59056 D0I2UH 44187006 IC50 = 3.7 nM T59056 D0I5NW 6540047 IC50 = 7 nM T59056 D0I9PA 25180306 IC50 = 154 nM T59056 D0J2WW 6539801 IC50 = 26 nM T59056 D0JE1I 9815923 IC50 = 1.8 nM T59056 D0K2DR 12050204 IC50 = 14 nM T59056 D0K3CE 6539800 IC50 = 3 nM T59056 D0K5KG 6540050 IC50 = 7 nM T59056 D0L2QD 45103910 IC50 = 22.91 nM T59056 D0L4NG 6540054 IC50 = 176 nM T59056 D0L8KL 11275595 IC50 = 12 nM T59056 D0LJ9D 46901783 IC50 = 796 nM T59056 D0M7FS 6539764 IC50 = 11 nM T59056 D0M9VK 11514098 IC50 = 218 nM T59056 D0MA9G 6540051 IC50 = 30 nM T59056 D0N1GH 11601068 IC50 = 2.9 nM T59056 D0N1PQ 11506923 IC50 = 6 nM T59056 D0N4VI 3021558 IC50 = 334 nM T59056 D0N5GZ 12229395 IC50 = 320 nM T59056 D0N8QD 15594569 IC50 > 1000 nM T59056 D0N9PY 6539773 IC50 = 79 nM T59056 D0NV7W 45103912 IC50 = 2.291 nM T59056 D0NX0M 6540049 IC50 = 2 nM T59056 D0O7TC 25180103 IC50 = 12 nM T59056 D0P1UO 45103914 IC50 = 25 nM T59056 D0PH1G 13688208 IC50 = 12.88 nM T59056 D0Q0BK 46901611 IC50 = 110 nM T59056 D0Q3CX 25034343 IC50 = 0.6 nM T59056 D0Q3JZ 6539774 IC50 = 248 nM T59056 D0Q5ZZ 25129117 IC50 = 53 nM T59056 D0Q6BJ 25034426 IC50 = 4.8 nM T59056 D0Q8KM 44206482 IC50 = 1.698 nM T59056 D0R0TE 11557864 IC50 = 12 nM T59056 D0RJ6S 11558270 IC50 = 15 nM T59056 D0S4KP 25034427 IC50 = 3.1 nM T59056 D0S4WQ 12229386 IC50 = 457 nM T59056 D0S8FV 44586852 IC50 = 7 nM T59056 D0T8JU 45103811 IC50 = 14 nM T59056 D0TM4K 6539817 IC50 = 13 nM T59056 D0U6IT 6539807 IC50 = 5 nM T59056 D0U7RR 6539768 IC50 = 171 nM T59056 D0V3YH 6539784 IC50 = 9 nM T59056 D0V6QN 45103915 IC50 = 117 nM T59056 D0V8CR 6539763 IC50 = 7 nM T59056 D0VL3R 25180303 IC50 = 29 nM T59056 D0W8IZ 45103809 IC50 = 5.754 nM T59056 D0WN9P 46901444 IC50 = 921 nM T59056 D0X0IH 77918 IC50 = 456 nM T59056 D0X1QS 6540053 IC50 = 13 nM T59056 D0Y0CT 6539819 IC50 = 3 nM T59056 D0Y3AV 25034346 IC50 = 5.1 nM T59056 D0Y5KX 46901443 IC50 = 406 nM T59056 D0YD9J 6539792 IC50 = 18 nM T59056 D0YS2F 6539776 IC50 = 27 nM T59056 D0Z3GX 46901784 IC50 = 331 nM T59056 D0Z4GR 4594970 IC50 = 22 nM T66396 D04AHQ 71721540 IC50 = 450 nM T66396 C3VRO9 44557921 IC50 > 10000 nM T66396 CX0R1K 53469059 IC50 = 3388 nM T66396 CV7C0D 53469060 IC50 = 776 nM T66396 COH62U 60097413 IC50 > 10000 nM T66396 C1MR8Q 60097495 IC50 > 2500 nM T66396 C7R0OL 71654743 IC50 < 300 nM T66396 CX4H6I 86583042 IC50 = 420 nM T66396 CVR43W 86583044 IC50 = 97 nM T66396 CA81UY 86583045 IC50 = 7300 nM T66396 C5LQG9 89769061 IC50 = 300 nM T66396 C28ADW 90655894 IC50 < 300 nM T66396 CPY8X5 90655895 IC50 < 300 nM T66396 C9KV8N 90655896 IC50 < 300 nM T66396 C5QC8E 118730408 IC50 = 3900 nM T66396 C4TXF2 118730409 IC50 = 290 nM T66396 CN2A9O 118730410 IC50 = 42 nM T66396 COF69K 118730411 IC50 = 5 nM T66396 CEJ1S6 118730412 IC50 = 12 nM T66396 CQ0T5Z 118730413 IC50 = 10 nM T66396 CF47CO 118730414 IC50 = 36 nM T66396 CEJ67D 118730415 IC50 = 42 nM T66396 C5SI6Q 118730416 IC50 = 240 nM T66396 CR0H9D 118730417 IC50 > 10000 nM T66396 CGDW48 118730418 IC50 = 1400 nM T66396 C23KFD 118730419 IC50 = 100 nM T66396 CJ9SA8 118730420 IC50 = 310 nM T66396 C0HK5A 118730421 IC50 = 610 nM T66396 C1Q0UN 118730422 IC50 > 50000 nM T66396 C1K0PE 118730423 IC50 > 50000 nM T66396 C2MD1Q 155513187 IC50 > 10000 nM T66396 D0T5VB 90655897 IC50 < 300 nM T74570 D0S5IR 86294073 IC50 > 30000 nM T74570 C0I8GC 14985965 IC50 > 100000 nM T74570 C2SOY1 46785920 IC50 > 30000 nM T74570 CFZ75O 46880148 IC50 > 30000 nM T74570 CL59YO 49852191 IC50 > 30000 nM T74570 C7ZUF5 49852192 IC50 > 30000 nM T74570 C6KX1V 49852195 IC50 > 30000 nM T74570 C3XQE2 52337837 IC50 > 100000 nM T74570 C4E1NK 57331209 IC50 > 50000 nM T74570 CGUA26 57331668 IC50 > 50000 nM T74570 CM1G2P 59568656 IC50 > 50000 nM T74570 C2D3HQ 60168069 IC50 > 100000 nM T74570 C9J0EH 71603917 IC50 > 100000 nM T74570 CU4CW1 121313969 IC50 > 100000 nM T30286 D0S9QA 132999 EC50 = 4280 nM T30286 D02AIN 122678117 IC50 > 32000 nM T30286 D06TKE 9796088 IC50 = 31.62 nM T30286 D0NR3V 65637 EC50 = 8570 nM T30286 C8LK1V 11317275 EC50 = 7230 nM T30286 CD34SB 15982534 IC50 > 100000 nM T30286 CV27NR 16015404 IC50 = 5011.87 nM T30286 CC2UO9 16015637 IC50 = 50118.72 nM T30286 CQ62LZ 16803385 IC50 = 19952.62 nM T30286 CY59DU 17616875 IC50 < 199526.23 nM T30286 CD3A1C 35579115 IC50 = 158.49 nM T30286 CV84AF 39734391 IC50 = 31622.78 nM T30286 CC50GL 39734394 IC50 = 1258.93 nM T30286 CL41FE 46206000 IC50 > 100000 nM T30286 C5GWN7 46937419 EC50 = 24940 nM T30286 CK9L3C 46939334 EC50 = 7140 nM T30286 C89JVN 46939418 EC50 = 70670 nM T30286 CL5D4G 46939499 EC50 = 31590 nM T30286 CO9LX7 46939500 EC50 = 135730 nM T30286 CU98ZN 53386723 IC50 = 3981.07 nM T30286 CDG90A 56658576 IC50 = 316.23 nM T30286 CK9BH7 56658685 IC50 > 199526.23 nM T30286 C40VQA 56662019 IC50 = 39810.72 nM T30286 CY76ZF 56662020 IC50 = 5011.87 nM T30286 C06MAF 56662154 IC50 = 19952.62 nM T30286 C36LWN 56662155 IC50 = 2511.89 nM T30286 CC67MA 56662156 IC50 > 199526.23 nM T30286 C91VWQ 56662157 IC50 = 3162.28 nM T30286 C41JXW 56665509 IC50 = 3981.07 nM T30286 C48YMD 56665613 IC50 > 199526.23 nM T30286 C5GPD3 56665614 IC50 > 199526.23 nM T30286 CLH3F2 56668937 IC50 = 316.23 nM T30286 CC41RK 56668938 IC50 = 794.33 nM T30286 CE87DY 56672420 IC50 = 794.33 nM T30286 CU8TA0 56672421 IC50 = 100000 nM T30286 CZMJ98 56672531 IC50 = 5011.87 nM T30286 CEBM89 56672532 IC50 > 199526.23 nM T30286 CE0LI2 56672533 IC50 = 158489.32 nM T30286 CBVO32 56675803 IC50 = 1584.89 nM T30286 C91FGR 56675804 IC50 = 794.33 nM T30286 CX5I9D 56675805 IC50 = 6309.57 nM T30286 C6GLB7 56675914 IC50 > 199526.23 nM T30286 CW4S7Z 56679123 IC50 = 5011.87 nM T30286 CE4H6B 56679227 IC50 > 199526.23 nM T30286 C7WCZ1 56679228 IC50 = 39810.72 nM T30286 C68OFP 56682419 IC50 = 79432.82 nM T30286 C2D3HQ 60168069 IC50 > 100000 nM T30286 CA07TC 71517197 IC50 > 33000 nM T30286 C1YK2E 122678192 IC50 > 32000 nM T30286 C0KMD3 155523506 EC50 = 3980 nM T30286 D0J0ZK 46937420 EC50 = 103780 nM T65005 D0S5IR 86294073 IC50 > 30000 nM T65005 CU98ZN 53386723 IC50 = 5011.87 nM T65005 C2D3HQ 60168069 IC50 > 100000 nM T09423 C4E1NK 57331209 IC50 > 10000 nM T09423 CM1G2P 59568656 IC50 > 10000 nM T09423 C9J0EH 71603917 IC50 > 100000 nM T39523 D05MQK 110635 IC50 > 10000 nM T39523 D0F8RA 2153 IC50 > 200000 nM T39523 D0Z7ZM 135398744 IC50 = 22000 nM T39523 D0SM0W 44591583 IC50 = 730 nM T39523 D0T5PO 5092 IC50 > 200000 nM T39523 D05VBJ 71295299 IC50 > 10000 nM T39523 D0WS3T 72706254 IC50 > 10000 nM T39523 D01QUF 9842576 Ki = 7900 nM T39523 C6I7EX 63761 IC50 = 6900 nM T39523 CX5HW2 376977 IC50 = 1500 nM T39523 CG7US1 680914 IC50 = 4680 nM T39523 CWU5J9 699904 IC50 = 7600 nM T39523 CXP6N7 806148 IC50 = 600 nM T39523 C5JN1M 895264 IC50 = 1290 nM T39523 CV58UI 959555 IC50 = 7980 nM T39523 C8JLO0 2243267 IC50 > 10000 nM T39523 CEVS38 2777384 IC50 = 6480 nM T39523 C7F0WA 2804210 IC50 = 3600 nM T39523 CK5R0M 2806991 IC50 = 2200 nM T39523 CZX6R8 2807179 IC50 = 5750 nM T39523 CS41AX 2915100 IC50 = 860 nM T39523 CGFN40 3008080 IC50 = 1040 nM T39523 CC3LA4 4672917 IC50 = 10 nM T39523 C5P0LU 4672918 IC50 = 10 nM T39523 CB40PM 6918356 IC50 = 1700 nM T39523 CR0NJ7 6918510 IC50 = 11000 nM T39523 COQP18 6918511 IC50 = 25000 nM T39523 CJ8EA9 6918641 IC50 = 60 nM T39523 C6G4QC 6918642 IC50 = 60 nM T39523 C1J5WZ 6918666 IC50 = 10 nM T39523 CI7K0P 6918667 IC50 = 10 nM T39523 CP1GO7 6918668 IC50 = 10 nM T39523 CH7QO4 6918791 IC50 = 20 nM T39523 CEBY83 6918792 IC50 = 3.9 nM T39523 C87WYR 6918795 IC50 = 20 nM T39523 CRGE51 6918796 IC50 = 20 nM T39523 CUP4M8 6918797 IC50 = 20 nM T39523 C0LRO8 6918798 IC50 = 40 nM T39523 C53ESK 6918799 IC50 = 50 nM T39523 CU1E0G 6918800 IC50 = 30 nM T39523 C36GKP 9813371 IC50 = 790 nM T39523 CD93RS 9813678 IC50 = 170 nM T39523 C1TU9E 9813679 IC50 = 2700 nM T39523 CQG16C 9834745 IC50 = 9500 nM T39523 CP9C4H 9835391 IC50 = 4800 nM T39523 CG0J5B 9835515 IC50 = 3700 nM T39523 C1NH4Q 9835516 IC50 = 600 nM T39523 C2VLX0 9835752 IC50 = 3080 nM T39523 CI1FX4 9835786 IC50 = 60 nM T39523 C6AMO1 9836267 IC50 = 60 nM T39523 CTU92B 9836268 IC50 = 210 nM T39523 C4J2XE 9836643 IC50 = 1700 nM T39523 C6HV9M 9836880 IC50 = 5900 nM T39523 C9NKL5 9856946 IC50 = 160 nM T39523 C18EZT 9857161 IC50 = 290 nM T39523 CG8ON7 9857246 IC50 = 980 nM T39523 CN1YU0 9857760 IC50 = 1500 nM T39523 CA23EP 9858103 IC50 = 60 nM T39523 C5DET1 9878144 IC50 = 3200 nM T39523 CA5MT8 9878456 IC50 = 160 nM T39523 C4R2UO 9878483 IC50 = 1400 nM T39523 C0Q5VN 9880010 IC50 = 5300 nM T39523 CWD1F6 9880288 IC50 = 960 nM T39523 CF7PS2 9899467 IC50 = 390 nM T39523 CJ47SK 9900486 IC50 = 120 nM T39523 CC05QE 9901606 IC50 = 2200 nM T39523 C6TC0L 9921876 IC50 = 2960 nM T39523 CBA29H 9922545 IC50 = 20 nM T39523 CKF4C2 9922691 IC50 = 1040 nM T39523 CTX25F 9924125 IC50 = 6850 nM T39523 C70AMC 9924305 IC50 = 140 nM T39523 CKI6N2 9924468 IC50 = 4 nM T39523 C6AZ5F 9924709 IC50 = 210 nM T39523 CNCL72 9942589 IC50 = 6600 nM T39523 CZY0V7 9942968 IC50 = 840 nM T39523 CF37NW 9943228 IC50 = 100 nM T39523 C84PKD 9943277 IC50 = 10 nM T39523 CA1S6U 9946483 IC50 = 130 nM T39523 CX1UV7 9946954 IC50 = 2130 nM T39523 C7OP5A 9947052 IC50 = 150 nM T39523 C9JVP5 9964901 IC50 = 4800 nM T39523 CRS0U5 9965532 IC50 = 10 nM T39523 CM76QK 9966726 IC50 = 870 nM T39523 CJO0X4 9966737 IC50 = 1800 nM T39523 CFP1Y5 9966830 IC50 = 6600 nM T39523 C0XJ1N 9966833 IC50 = 1050 nM T39523 C9NKY4 9967652 IC50 = 150 nM T39523 CI6AX1 9968005 IC50 = 1630 nM T39523 C7PCS8 9968050 IC50 = 4600 nM T39523 CFB48Q 9968370 IC50 = 1240 nM T39523 CU73AJ 9968471 IC50 = 1620 nM T39523 C0AP8O 9969020 IC50 = 160 nM T39523 C12LED 10109572 IC50 = 400 nM T39523 C2PBD6 10131447 IC50 = 50 nM T39523 C8NT0W 10131621 IC50 = 140 nM T39523 CJ24HR 10132715 IC50 = 200 nM T39523 C5HC2X 10182563 IC50 = 40 nM T39523 C3GN8K 10200432 IC50 = 10 nM T39523 CFGO46 10221904 IC50 = 10 nM T39523 C1XL2R 10247726 IC50 = 8000 nM T39523 CQ61CV 10268304 IC50 = 30 nM T39523 C1QU2B 10268305 IC50 = 30 nM T39523 CH9C4K 10269859 IC50 = 1370 nM T39523 CR92JY 10270352 IC50 = 40 nM T39523 C7CHR0 10270536 IC50 = 20 nM T39523 CIA5D7 10685727 IC50 = 2950 nM T39523 C8UHE3 10717022 IC50 = 15000 nM T39523 C28FLE 10762239 IC50 = 28000 nM T39523 C5BA7H 10802745 IC50 = 5690 nM T39523 C24LPM 10810360 IC50 = 22000 nM T39523 CT2F6P 10835916 IC50 = 13000 nM T39523 CBA38X 11513431 IC50 = 14 nM T39523 CQ8Y6L 11793138 IC50 = 21000 nM T39523 C7E8QN 11796403 IC50 = 14000 nM T39523 C1B4XD 11992634 IC50 > 2000 nM T39523 CPX16N 11993169 IC50 > 2000 nM T39523 CC3Q2L 12466688 IC50 = 7300 nM T39523 CQM6H9 12700219 IC50 = 2200 nM T39523 C9WKV0 14531504 IC50 = 370 nM T39523 CVR73F 15549302 IC50 = 7700 nM T39523 CQT1H8 17834549 IC50 = 6500 nM T39523 CG4D0L 18436679 IC50 = 18 nM T39523 CS6HD4 18967579 IC50 = 5200 nM T39523 C9M0ZA 21483258 IC50 = 2200 nM T39523 CY06TV 21920178 IC50 = 560 nM T39523 CL30BY 21920189 IC50 = 20 nM T39523 C15BGX 21920191 IC50 = 150 nM T39523 CMZ5G9 21920202 IC50 = 90 nM T39523 CIB31Y 21920218 IC50 = 60 nM T39523 CL4R5H 21920232 IC50 = 550 nM T39523 C68RSV 21920245 IC50 = 30 nM T39523 C76SHB 21920252 IC50 = 80 nM T39523 CA2LZ9 21920253 IC50 = 4000 nM T39523 C7RK1W 21920272 IC50 = 260 nM T39523 CH7N9S 21920275 IC50 = 80 nM T39523 CBPD46 21920277 IC50 = 120 nM T39523 C90EXZ 21920288 IC50 = 60 nM T39523 CWHX89 21920307 IC50 = 930 nM T39523 CIRD07 21920317 IC50 = 1900 nM T39523 CW5MP2 21920319 IC50 = 3900 nM T39523 CEDO71 21920329 IC50 = 700 nM T39523 C18YNU 21920341 IC50 = 470 nM T39523 C0JOK1 21920350 IC50 = 1300 nM T39523 CRN3H8 21920369 IC50 = 470 nM T39523 CV04DH 21920370 IC50 = 5700 nM T39523 C78SFX 21920385 IC50 = 5600 nM T39523 CFAQ86 22343616 IC50 = 180 nM T39523 C4S6VD 23654252 IC50 > 50000 nM T39523 CA3H8C 24100795 IC50 = 580 nM T39523 C9WGI4 24802717 IC50 = 3345 nM T39523 CL38GE 24905352 IC50 = 3230 nM T39523 CW1PC2 24970381 IC50 = 7020 nM T39523 CRW7P6 25020172 IC50 = 9300 nM T39523 CF3UQ7 25020175 IC50 = 5070 nM T39523 CC7A3M 25020230 IC50 = 1700 nM T39523 CHF6P7 25020232 IC50 = 1690 nM T39523 C2AG8Z 25020234 IC50 = 480 nM T39523 CNJ09P 25020295 IC50 = 5330 nM T39523 C93DZI 25147798 IC50 > 50000 nM T39523 CPC08B 25179287 IC50 > 50000 nM T39523 COB03R 25179478 IC50 = 17000 nM T39523 CDE2I7 25229546 IC50 = 510 nM T39523 CICF39 42629702 IC50 = 2318 nM T39523 CM3X9S 42629827 IC50 = 332 nM T39523 CQN26J 42629945 IC50 = 542 nM T39523 C6O5FX 42630062 IC50 = 2930 nM T39523 C71ZNR 42630180 IC50 = 266 nM T39523 C4RHY0 42630191 IC50 > 100000 nM T39523 CT6RS9 42630192 IC50 > 10000 nM T39523 CYZL43 42630317 IC50 > 10000 nM T39523 CH42OZ 42630318 IC50 > 10000 nM T39523 C7X5AH 42630437 IC50 > 10000 nM T39523 CW8OB3 44243146 Ki > 10000 nM T39523 C13HPW 44393651 IC50 = 1520 nM T39523 CJ6GB5 44393709 IC50 = 20 nM T39523 CE8TU4 44393929 IC50 = 5900 nM T39523 C8U2DW 44393934 IC50 = 7500 nM T39523 CQP01D 44393950 IC50 = 1310 nM T39523 C6A7JK 44393959 IC50 = 1650 nM T39523 CU1CQ8 44394047 IC50 = 10 nM T39523 CTX1E5 44394060 IC50 = 230 nM T39523 C9UBW7 44394109 IC50 = 2660 nM T39523 CL56ZH 44394110 IC50 = 6540 nM T39523 CBL2J9 45263650 IC50 > 10000 nM T39523 C5IMB2 46239424 Ki > 10000 nM T39523 CKR9P7 46239425 Ki > 10000 nM T39523 C3P2IN 46933992 IC50 >= 75000 nM T39523 CHA5Z0 49821469 IC50 > 1000 nM T39523 C1AYP0 49821627 IC50 > 500 nM T39523 C85AXR 49821714 IC50 > 1000 nM T39523 C0B8JE 49843464 Ki = 2472 nM T39523 CMN05G 50901953 Ki = 11085 nM T39523 CPL5E6 50902114 Ki = 5536 nM T39523 CAD40F 50902119 Ki = 6935 nM T39523 CD98UC 50902202 Ki = 10114 nM T39523 CXB85R 50902203 Ki = 7499 nM T39523 C9QLF2 50902206 Ki = 3760 nM T39523 CH2Z1E 50902289 Ki = 6119 nM T39523 C4HJL2 50902291 Ki = 5982 nM T39523 C7EQ9Y 50902548 Ki = 613 nM T39523 C6A1IU 50902549 Ki = 243 nM T39523 CVM28N 50902550 Ki = 269 nM T39523 CN1P7Q 50902632 Ki = 550 nM T39523 C3Y2AV 50903255 Ki = 3701 nM T39523 CGF65A 54670110 IC50 > 30000 nM T39523 C90ZLC 54670399 IC50 = 1170 nM T39523 CC9Z2M 54908813 IC50 = 3300 nM T39523 C4TGL7 56648496 IC50 = 1300 nM T39523 CH6C3L 56648679 IC50 = 1170 nM T39523 CCY79V 56648680 IC50 = 824 nM T39523 CNE96P 56648857 IC50 = 919 nM T39523 CX86AQ 56648859 IC50 = 1340 nM T39523 C0YD3P 56928304 IC50 = 60 nM T39523 C8RO6A 56929788 IC50 = 13 nM T39523 CND81R 56968371 IC50 = 6100 nM T39523 CY7AO0 56968372 IC50 = 1800 nM T39523 CV6P2I 57385525 IC50 = 33370 nM T39523 CUS7R9 57385526 IC50 = 12340 nM T39523 CB17SC 57385767 IC50 = 5170 nM T39523 CH75PT 57385768 IC50 = 2630 nM T39523 CYE1Z4 57386041 IC50 = 7310 nM T39523 C7EB5V 57386043 IC50 = 14070 nM T39523 CK81XA 57386556 IC50 = 3200 nM T39523 C2ZD7G 57390975 IC50 = 66 nM T39523 CHB1V2 57390976 IC50 = 82 nM T39523 CO75IQ 57390977 IC50 = 104 nM T39523 C6EI3A 57390978 IC50 = 24 nM T39523 C5CLS9 57390979 IC50 = 96 nM T39523 C61WPI 57390980 IC50 = 300 nM T39523 CDHJ84 57390991 IC50 = 206 nM T39523 C6W8KX 57390992 IC50 = 212 nM T39523 CES36G 57390993 IC50 > 1000 nM T39523 C01JFV 57390994 IC50 = 686 nM T39523 CODM26 57390995 IC50 = 34 nM T39523 CD52CA 57391118 IC50 > 2000 nM T39523 C68NJH 57392756 IC50 > 5000 nM T39523 CJPE69 57392757 IC50 = 29 nM T39523 CN85ZR 57392758 IC50 = 27 nM T39523 C2A5RM 57392759 IC50 = 34 nM T39523 C0F7ON 57392760 IC50 = 25 nM T39523 CLV6C2 57392761 IC50 = 86 nM T39523 C5IAB9 57392762 IC50 = 105 nM T39523 CI9K4B 57392763 IC50 = 151 nM T39523 CT67RF 57392774 IC50 > 1000 nM T39523 CPNH58 57392775 IC50 = 192 nM T39523 CJV0C8 57392776 IC50 = 17 nM T39523 C89ZVD 57392777 IC50 = 18 nM T39523 C0LZ1P 57392778 IC50 = 59 nM T39523 CG3DF1 57392948 Ki > 10000 nM T39523 CD3QS0 57394488 IC50 = 823 nM T39523 C8DIO6 57394489 IC50 = 1070 nM T39523 CPA7C8 57394490 IC50 = 179 nM T39523 C52PKN 57394491 IC50 = 20 nM T39523 C0G9QL 57394492 IC50 = 188 nM T39523 CNS3R5 57394502 IC50 = 90 nM T39523 C8HNQ3 57394503 IC50 = 712 nM T39523 C85UHM 57394504 IC50 = 165 nM T39523 C7SX3Y 57394505 IC50 = 33 nM T39523 CHE68W 57394506 IC50 = 868 nM T39523 C1V0IE 57394507 IC50 = 44 nM T39523 C0F6OX 57394508 IC50 = 12 nM T39523 CE36TV 57394695 Ki > 10000 nM T39523 CJ6E9Q 57396249 IC50 = 200 nM T39523 CI8S6J 57396252 IC50 = 18 nM T39523 CZ3V0H 57396253 IC50 = 32 nM T39523 CT9XE7 57398056 IC50 > 1000 nM T39523 COQJ51 57398057 IC50 = 10 nM T39523 CFB2P9 57399706 IC50 = 46 nM T39523 C2B1AF 57399707 IC50 = 29 nM T39523 C7MWD1 57399708 IC50 = 49 nM T39523 C8UZ1R 57399715 IC50 = 266 nM T39523 CO3AG1 57399716 IC50 = 18 nM T39523 CX27HZ 57401470 IC50 = 124 nM T39523 C8QU1A 57401471 IC50 = 71 nM T39523 C0FW5U 57401478 IC50 = 39 nM T39523 C1WS7F 57403204 IC50 = 22 nM T39523 C0KL7Y 57403205 IC50 = 94 nM T39523 C2UX3A 57403206 IC50 > 1000 nM T39523 CP0L9U 57403207 IC50 = 176 nM T39523 CX4M5I 57403214 IC50 = 767 nM T39523 COYT07 57403215 IC50 = 2380 nM T39523 C0C6TW 57403216 IC50 > 1000 nM T39523 C3D1OC 57403217 IC50 = 317 nM T39523 CCA5S3 57403218 IC50 = 178 nM T39523 C6DA0M 57403219 IC50 > 1000 nM T39523 CJ6TS1 57403220 IC50 = 88 nM T39523 CB4PT8 57403221 IC50 = 20 nM T39523 CPA3D1 57403394 Ki > 10000 nM T39523 C4XMB6 58547809 IC50 > 30000 nM T39523 CEB3G9 58547814 IC50 > 30000 nM T39523 C08QVG 58547833 IC50 > 30000 nM T39523 CFVG67 58547863 IC50 > 30000 nM T39523 CYZA38 58548077 IC50 > 30000 nM T39523 C93TFZ 59788598 IC50 = 1880 nM T39523 CU9GQ0 70681149 Ki = 4596 nM T39523 CI9G8L 70683261 Ki = 3770 nM T39523 C6BN5J 70685361 Ki = 507 nM T39523 CF6O3T 70687501 Ki = 4599 nM T39523 CZ7B8O 70688228 IC50 = 880 nM T39523 C4P0XT 71092344 IC50 = 660 nM T39523 C6DAG4 71092519 IC50 = 3460 nM T39523 C2HGI7 71153408 IC50 > 10000 nM T39523 C9GR3L 71153436 IC50 = 1910 nM T39523 C68SDB 71719394 IC50 = 3162.28 nM T39523 CSR5Z9 71727398 IC50 = 1070 nM T39523 CZ3X1I 71727503 IC50 = 539 nM T39523 CO94RY 71727504 IC50 > 1000 nM T39523 C4X1MC 71727505 IC50 = 521 nM T39523 C85ODL 71727506 IC50 = 46 nM T39523 CDE7W9 71727609 IC50 > 1000 nM T39523 CLU28C 71727610 IC50 > 5000 nM T39523 C2I7RY 71727611 IC50 > 5000 nM T39523 CT6CN3 71727612 IC50 > 5000 nM T39523 C62UOR 71727613 IC50 > 5000 nM T39523 C42SID 71727614 IC50 = 1050 nM T39523 CQ3JC7 71727615 IC50 > 1000 nM T39523 C15JYG 71727720 IC50 > 5000 nM T39523 C7BTQ8 71727721 IC50 > 5000 nM T39523 CC8SE6 71727722 IC50 > 5000 nM T39523 CS3BJ5 71727841 IC50 > 5000 nM T39523 C6R0XV 76313636 IC50 = 15250 nM T39523 CIXB87 80053866 IC50 = 3800 nM T39523 CJ1EB2 85839481 IC50 = 3970 nM T39523 CY34OK 86280445 IC50 = 42 nM T39523 C4BD5F 91667427 IC50 = 4.4 nM T39523 C45QVJ 91668196 IC50 = 3.3 nM T39523 C1JPD6 91844700 IC50 = 4200 nM T39523 CQCA74 101886683 IC50 = 720 nM T39523 C2L1SH 101886684 IC50 = 990 nM T39523 COZ0H2 101886685 IC50 = 1010 nM T39523 CJD4X0 101886686 IC50 = 1470 nM T39523 CE41HT 101886687 IC50 = 5450 nM T39523 C8UIX0 101886688 IC50 = 2140 nM T39523 CMRP31 101886690 IC50 = 2100 nM T39523 C4LQ7R 101891513 IC50 = 2 nM T39523 CYQ74R 118479645 IC50 > 10000 nM T39523 C8N4FR 118719983 IC50 = 160 nM T39523 C1DN6I 118719984 IC50 = 1100 nM T39523 COX37C 118719985 IC50 = 310 nM T39523 C8O1QW 118719986 IC50 = 6800 nM T39523 CO1XA7 118719987 IC50 = 5000 nM T39523 C9NCB0 118719988 IC50 = 150 nM T39523 CQTX25 118719989 IC50 = 740 nM T39523 CIH74Z 118719990 IC50 = 11000 nM T39523 CC4IU3 118719991 IC50 = 6500 nM T39523 CC48FZ 118719992 IC50 > 1000 nM T39523 C5FOB6 118719993 IC50 = 2600 nM T39523 CX92KJ 118719994 IC50 = 98 nM T39523 COLJ03 118719995 IC50 = 30 nM T39523 C0Z3GQ 118719996 IC50 = 45 nM T39523 CY2NS6 118719997 IC50 = 67 nM T39523 C1WC8D 118719998 IC50 = 4.2 nM T39523 C1UBR0 118719999 IC50 = 19 nM T39523 CB29OG 118720000 IC50 = 7.3 nM T39523 CM6ZP8 118720001 IC50 = 39 nM T39523 C8HP5T 118720002 IC50 = 5.6 nM T39523 CSIF10 118720003 IC50 = 380 nM T39523 C1WE3G 118720004 IC50 = 5 nM T39523 CZYT12 118720005 IC50 = 4.9 nM T39523 CW41JN 118720006 IC50 = 2.3 nM T39523 CU56DJ 118720007 IC50 = 1 nM T39523 CD6U4P 118720008 IC50 = 12 nM T39523 C60JDU 118723252 IC50 = 8770 nM T39523 CY7N6M 118723253 IC50 = 9270 nM T39523 CB79OS 118723255 IC50 = 3200 nM T39523 CY50ZX 118723256 IC50 = 6180 nM T39523 CV0MP6 118723257 IC50 = 2880 nM T39523 CJYZ53 118723745 IC50 = 1600 nM T39523 C2WHE3 118723751 IC50 = 4270 nM T39523 CJY41B 118723752 IC50 = 124000 nM T39523 C9U6TB 118724077 IC50 = 290 nM T39523 CUQ6W2 118724078 IC50 = 88 nM T39523 CNP0Z2 118724079 IC50 > 1000 nM T39523 CVH9Z2 118724080 IC50 > 1000 nM T39523 CYC1O5 118724081 IC50 > 1000 nM T39523 CXK30G 118724082 IC50 = 2300 nM T39523 CP0X8J 118724083 IC50 = 61 nM T39523 CWRL26 118724084 IC50 = 41 nM T39523 CXQC01 118724085 IC50 > 1000 nM T39523 C5B7AW 118724086 IC50 = 630 nM T39523 CNM6F3 118724087 IC50 = 60 nM T39523 CH4L6O 118724088 IC50 = 25 nM T39523 CCZ6W9 118724089 IC50 = 8.7 nM T39523 C40AXS 118724090 IC50 = 2.1 nM T39523 CKG08X 118724091 IC50 = 3.9 nM T39523 C3OR6T 118724092 IC50 = 1.1 nM T39523 CM6XW1 118724093 IC50 = 0.68 nM T39523 C46LFG 118724094 IC50 = 1.2 nM T39523 CYM21X 118724095 IC50 = 0.32 nM T39523 C1H6SK 118729734 IC50 = 2900 nM T39523 CML97J 118729735 IC50 = 1400 nM T39523 CM8EO1 118729736 IC50 = 370 nM T39523 C4E3UH 118729737 IC50 = 4700 nM T39523 CSV23W 118729738 IC50 = 1500 nM T39523 CY95EQ 118729739 IC50 = 2600 nM T39523 CDHC56 118729740 IC50 = 300 nM T39523 CEKR01 118729741 IC50 = 430 nM T39523 CBJ24Z 118729742 IC50 = 2300 nM T39523 CFK03G 118729743 IC50 = 2100 nM T39523 C3ETW0 118729744 IC50 = 1300 nM T39523 CL23ZS 118729745 IC50 = 12 nM T39523 CUW3D1 118729746 IC50 = 6.4 nM T39523 C1UL3B 118729747 IC50 = 4.6 nM T39523 C72ATF 118729748 IC50 = 7.6 nM T39523 C59LGI 118729749 IC50 = 190 nM T39523 CPQN92 118729750 IC50 = 170 nM T39523 C5MI9E 118729751 IC50 = 6.8 nM T39523 CE5ON1 118729752 IC50 = 20 nM T39523 CX0W4F 118729753 IC50 = 5.1 nM T39523 CB1DX3 118729754 IC50 = 15 nM T39523 CC41IT 118729755 IC50 = 8.4 nM T39523 CB2DX0 118729756 IC50 = 8.1 nM T39523 CB40SN 118729757 IC50 = 1.5 nM T39523 C4HI1Q 118729758 IC50 = 2.7 nM T39523 CKBG19 118729759 IC50 = 1.4 nM T39523 CS6M9C 122193679 IC50 > 100000 nM T39523 CACJ46 132489333 IC50 > 10000 nM T39523 C2P1IU 134129996 IC50 > 100000 nM T39523 CLE03O 134130328 IC50 > 100000 nM T39523 CSN6J0 134130563 IC50 > 100000 nM T39523 C0A1CZ 134131162 IC50 > 100000 nM T39523 C3R8SE 135457869 IC50 > 10000 nM T39523 CJS37E 135482260 IC50 = 3.5 nM T39523 CHDC83 135566745 IC50 > 10000 nM T39523 C9IJK1 135566935 IC50 = 1800 nM T39523 C3PO9K 135856789 IC50 = 440 nM T39523 C3M7VF 135856791 IC50 = 240 nM T39523 CAO3U7 135856794 IC50 = 6400 nM T39523 CTX54Z 135896326 IC50 > 10000 nM T39523 CD9E1F 135948887 IC50 = 1.3 nM T39523 C2FW0D 135981181 IC50 = 14 nM T39523 CJM3W6 135981182 IC50 = 16 nM T39523 C12UMG 136059728 IC50 > 1000 nM T39523 CRP24A 136087045 IC50 = 17900 nM T39523 C7SUX4 136087050 IC50 = 51200 nM T39523 C8UF7G 136087052 IC50 > 100000 nM T39523 C21FVA 136180322 IC50 > 10000 nM T39523 C8TQ7A 136217455 IC50 > 100000 nM T39523 C0KGW7 136230107 IC50 = 89 nM T39523 C1O2YF 136230108 IC50 = 93 nM T39523 CEJ34Q 136230109 IC50 = 3 nM T39523 C4Y6KS 136230111 IC50 = 75 nM T39523 CE4HQ5 136230157 IC50 = 31 nM T39523 CH5SF7 136230158 IC50 = 27 nM T39523 CI1W8Q 136230159 IC50 = 12 nM T39523 C8HNC5 136230160 IC50 = 104 nM T39523 C1PIQ4 136230176 IC50 = 73 nM T39523 C20PEA 136230178 IC50 = 45 nM T39523 C2AGJ6 136230179 IC50 = 53 nM T39523 C4Q3WN 136230180 IC50 = 71 nM T39523 CJ80XF 136230186 IC50 = 81 nM T39523 CN0HJ2 136230187 IC50 = 33 nM T39523 CO3DY1 136230188 IC50 = 32 nM T39523 CEPN61 136230189 IC50 = 18 nM T39523 C7FI5A 136230190 IC50 = 24 nM T39523 CDMI24 136230191 IC50 = 68 nM T39523 C4NMD5 136236286 IC50 = 55 nM T39523 CE30VQ 136236287 IC50 = 80 nM T39523 C5YXS9 136236288 IC50 = 77 nM T39523 CE0RJ7 136244191 IC50 = 8 nM T39523 C8JV5W 136244192 IC50 = 18 nM T39523 C6P9CK 136244193 IC50 = 11 nM T39523 CHU6X8 136244194 IC50 = 7 nM T39523 CV7D0S 136244195 IC50 = 106 nM T39523 CZP75Q 136244196 IC50 = 12 nM T39523 CWC6B4 136244198 IC50 = 30 nM T39523 CS2MF4 136244248 IC50 = 17 nM T39523 COQP79 136244250 IC50 = 80 nM T39523 CL21TN 136254165 IC50 = 47 nM T39523 CP8X1D 136254166 IC50 = 46 nM T39523 CGE6L9 136254167 IC50 = 9 nM T39523 C9Q2ZK 136254168 IC50 = 4 nM T39523 C7ORL8 136254169 IC50 = 23 nM T39523 CG24NK 136254170 IC50 = 16 nM T39523 C2F3JC 136254171 IC50 = 35 nM T39523 CEX4G5 136254172 IC50 = 12 nM T39523 C4SB9K 136254173 IC50 = 66 nM T39523 CH0Z9S 136254174 IC50 = 88 nM T39523 CI2VF8 136254175 IC50 = 125 nM T39523 CMYE58 136254176 IC50 = 18 nM T39523 C85RTY 136254177 IC50 = 35 nM T39523 C4X9ZM 136254178 IC50 = 38 nM T39523 C6GWA0 136254179 IC50 = 15 nM T39523 COE54I 136254180 IC50 = 25 nM T39523 CXN6R3 136254181 IC50 = 101 nM T39523 CR5WY9 136254182 IC50 = 39 nM T39523 C24XKG 136254183 IC50 = 46 nM T39523 CSX2F1 136254184 IC50 = 14 nM T39523 CY9JG0 136254185 IC50 = 31 nM T39523 C6KYD7 137700754 IC50 = 4830 nM T39523 CM3UF7 137700779 IC50 > 20000 nM T39523 CPTE92 138319693 IC50 > 32000 nM T39523 C2QLX3 138393292 IC50 > 5000 nM T39523 CMW20N 141737696 IC50 > 4000 nM T39523 C8HEG7 141737705 IC50 > 3000 nM T39523 C5CL3K 145964282 IC50 = 3200 nM T39523 C0IC6F 145964309 IC50 = 33600 nM T39523 CCM4E7 145964412 IC50 > 200000 nM T39523 CEV2C0 145965057 IC50 = 10500 nM T39523 CZF69G 145966063 IC50 = 48900 nM T39523 C1H4RT 145966342 IC50 = 92900 nM T39523 C4JR7O 145967554 IC50 > 200000 nM T39523 C6YXM2 145968230 IC50 = 7300 nM T39523 CK2Q1M 145972042 IC50 > 200000 nM T39523 CXY3H9 145973870 IC50 = 140900 nM T39523 CY2R1M 145974127 IC50 > 200000 nM T39523 CC7HN2 145974174 IC50 > 100000 nM T39523 CZEW75 145974259 IC50 = 115900 nM T39523 CL0ZP8 145974645 IC50 = 3800 nM T39523 C0JQ3V 145974692 IC50 > 200000 nM T39523 CLV25P 145974711 IC50 = 52800 nM T39523 CNBC60 145975232 IC50 > 200000 nM T39523 C6W7RB 145975941 IC50 = 11700 nM T39523 CS1V9B 145976314 IC50 = 89300 nM T39523 CN61GR 145977095 IC50 = 69800 nM T39523 CD09US 145977528 IC50 = 56100 nM T39523 CTZ6O9 145977634 IC50 = 8100 nM T39523 CZ50HJ 145977998 IC50 = 27600 nM T39523 CK1BR0 145978345 IC50 > 100000 nM T39523 CKOT32 145978829 IC50 = 9500 nM T39523 CZC61L 145978996 IC50 > 200000 nM T39523 C0JRK5 145980304 IC50 > 200000 nM T39523 CV7G5F 145981927 IC50 = 19750 nM T39523 C7BP2S 145981946 IC50 > 200000 nM T39523 C42VHC 145982018 IC50 = 9060 nM T39523 C5RCY6 145982932 IC50 > 200000 nM T39523 CT1L8E 145986656 IC50 = 54280 nM T39523 C1TU2D 145986784 IC50 = 5070 nM T39523 CAS90U 145986925 IC50 = 37590 nM T39523 C3SV8R 145987119 IC50 > 200000 nM T39523 CM6P3Z 145987468 IC50 = 96320 nM T39523 C0ODP3 145988021 IC50 > 200000 nM T39523 C25WHX 145988690 IC50 = 41150 nM T39523 C35GWH 145989417 IC50 = 19960 nM T39523 CY75SD 145989570 IC50 > 200000 nM T39523 CUK86E 145989957 IC50 = 7760 nM T39523 CV9BP4 145990259 IC50 > 200000 nM T39523 C6NHE1 145990687 IC50 > 200000 nM T39523 COSL82 145992781 IC50 > 200000 nM T39523 C8CSM5 145992787 IC50 > 200000 nM T39523 CG5E3A 145993704 IC50 > 200000 nM T39523 CI7H3T 145994146 IC50 > 200000 nM T39523 CHJ79V 145997874 IC50 = 620 nM T39523 CM7TX2 148279038 IC50 > 100000 nM T39523 CL8CU6 155521936 IC50 > 200000 nM T39523 CT85RG 155530589 IC50 > 200000 nM T39523 D00MBG 2921148 IC50 = 90 nM T39523 D09RKU 46239428 Ki > 10000 nM T39523 D0D6MC 1150897 IC50 > 200000 nM T39523 D0R6MT 3758 IC50 = 85600 nM T83202 D0E6XR 3062316 IC50 > 20000 nM T83202 D0R0MW 5329102 IC50 = 131.3 nM T83202 D01NEC 51042438 IC50 = 339 nM T83202 D02ZQS 16095342 IC50 = 132 nM T83202 D0E3TC 44259 IC50 = 0.09 nM T83202 D0MS3Z 16725726 IC50 = 1260 nM T83202 D03BNU 59604787 IC50 > 10000 nM T83202 D02GEJ 5326976 IC50 = 10280 nM T83202 D0T3ME 156422 IC50 > 30000 nM T83202 C4RUV5 5329453 IC50 = 2100 nM T83202 CJO47T 9948405 IC50 > 10000 nM T83202 CV8I5X 9999342 IC50 > 10000 nM T83202 C5TQ7X 10247543 IC50 > 10000 nM T83202 C2WQ8M 10473563 IC50 > 10000 nM T83202 CLZK93 11189172 IC50 = 740 nM T83202 CM6DO0 11233873 IC50 = 3100 nM T83202 CRG03D 11245934 IC50 = 44 nM T83202 C0OZW2 11247002 IC50 = 620 nM T83202 CN16LZ 11269477 IC50 = 1100 nM T83202 COW1S8 11360518 IC50 = 1410 nM T83202 C9UI3O 11373846 IC50 = 780 nM T83202 CONW29 11453116 IC50 = 1950 nM T83202 C7IOJ0 11548023 IC50 = 398 nM T83202 CACS26 11561968 Ki > 2000 nM T83202 CJS28X 11641672 IC50 = 510 nM T83202 CU0E8O 11690457 Ki > 2000 nM T83202 COH3C4 11697546 IC50 = 5300 nM T83202 C5ISQ9 11751266 IC50 = 90 nM T83202 C3YRU7 15295578 IC50 = 810 nM T83202 C7Z4LV 16095343 IC50 = 35 nM T83202 CQK6C4 16099866 IC50 > 10000 nM T83202 CG6D4M 23647319 IC50 > 10000 nM T83202 CY8Z7X 23647330 IC50 > 10000 nM T83202 C4XD8H 23647348 IC50 > 10000 nM T83202 C2UOE0 24766030 IC50 > 50000 nM T83202 CY8L7E 24896769 IC50 > 10000 nM T83202 CW2MV8 25023720 IC50 = 13 nM T83202 CPB4S2 25023721 IC50 = 71 nM T83202 CSM1R7 25023724 IC50 = 251 nM T83202 C4DF8X 25023725 IC50 = 1259 nM T83202 CXFQ18 25023726 IC50 = 1 nM T83202 C13MHS 25023727 IC50 = 6 nM T83202 C1JEU6 25023729 IC50 = 790 nM T83202 C14NAT 25023731 IC50 = 500 nM T83202 C81XKW 25023732 IC50 = 1560 nM T83202 CFH80B 25023733 IC50 = 1990 nM T83202 CR8JP7 25023735 IC50 = 1580 nM T83202 C4W7LY 25023736 IC50 = 2510 nM T83202 CA6QU5 25023737 IC50 = 500 nM T83202 CLFM35 25206064 IC50 = 780 nM T83202 CLW80F 44160269 IC50 = 11000 nM T83202 CK73NR 44219749 IC50 > 50000 nM T83202 COPG94 44427519 IC50 > 10000 nM T83202 C4WRN5 44541014 IC50 = 45.9 nM T83202 C3VRO9 44557921 IC50 > 10000 nM T83202 CCL85F 44575073 IC50 > 50000 nM T83202 CJX06P 44575126 IC50 > 50000 nM T83202 CE8FC7 44575127 IC50 > 50000 nM T83202 C28QLM 44605035 IC50 > 50000 nM T83202 C75XHS 44605037 IC50 > 50000 nM T83202 CC95PQ 45375865 IC50 > 50000 nM T83202 CEOQ27 45375866 IC50 > 50000 nM T83202 C96BNW 46179972 IC50 > 50000 nM T83202 CO3P0J 46866604 IC50 < 50000 nM T83202 CJOM49 46880136 IC50 = 9710 nM T83202 C1NKE3 46905987 IC50 = 1900 nM T83202 CQ3KU9 50899556 IC50 = 2100 nM T83202 C8CGM9 51346966 IC50 = 568 nM T83202 CEQN27 52936621 Ki > 1000 nM T83202 C3LB5V 52941849 IC50 = 3400 nM T83202 CW2X5E 52944268 IC50 = 560 nM T83202 C9PX2J 52945752 IC50 = 220 nM T83202 CL4ED3 52945753 IC50 = 1100 nM T83202 CIR3Q0 52947964 IC50 > 10000 nM T83202 C8NA4L 53384644 IC50 > 30000 nM T83202 CPC5D2 56603995 IC50 = 2510 nM T83202 CEBQ15 56604005 IC50 = 251 nM T83202 CFP56A 56604013 IC50 = 3980 nM T83202 CE8T5V 57393795 IC50 = 1181 nM T83202 C1MR8Q 60097495 IC50 > 1000 nM T83202 CUJ28O 67112053 IC50 = 699 nM T83202 C2ZJC1 67113434 IC50 = 272 nM T83202 CV63UL 67240318 IC50 > 5000 nM T83202 C1IEJ2 70789254 IC50 = 63000 nM T83202 C8T7ZP 70789255 IC50 = 13000 nM T83202 C0DL3F 72698602 IC50 < 1 nM T83202 C4X7SD 122192466 IC50 > 10000 nM T83202 C2LAM7 126591927 IC50 = 311 nM T83202 CO47QJ 133054002 IC50 = 20 nM T83202 C8GQD5 137636872 IC50 = 5.4 nM T83202 C28QUP 137652864 IC50 > 10000 nM T83202 CC73PA 138911338 IC50 = 131 nM T83202 CSU93V 155077019 IC50 = 32 nM T83202 C2MD1Q 155513187 IC50 > 10000 nM T83202 CL5DR0 155525783 IC50 = 48 nM T83202 D01YWE 25207521 IC50 = 290 nM T83202 D09PTP 57325421 IC50 = 61 nM T83202 D0W7TU 947057 IC50 = 34900 nM T83202 D0Y0BK 11524144 IC50 = 210 nM T46781 D00FGR 3599 IC50 > 100000 nM T46781 D04XGT 31593 IC50 > 100000 nM T46781 D05EAM 4735 IC50 > 100000 nM T46781 D0E6XR 3062316 IC50 = 6485 nM T46781 D0K8KX 5280343 IC50 = 910 nM T46781 D0R0MW 5329102 IC50 = 1500 nM T46781 D00LGR 56839178 IC50 = 12.4 nM T46781 D02RJY 11442891 Ki = 79 nM T46781 D02UFQ 11620908 IC50 = 1700 nM T46781 D02XNW 5494449 Ki = 1.8 nM T46781 D03HUX 49792852 IC50 > 10000 nM T46781 D05PZB 135398495 IC50 = 2.7 nM T46781 D08HOM 46207586 IC50 = 2 nM T46781 D0A1AQ 5329099 IC50 = 35 nM T46781 D0A5MC 11712649 IC50 = 4000 nM T46781 D0CY1B 6420138 Ki = 9.2 nM T46781 D0E3TC 44259 IC50 = 1 nM T46781 D0E5XA 11569967 IC50 = 54 nM T46781 D0EJ3B 24856041 IC50 = 4 nM T46781 D0IQ0Z 46885626 Ki = 0.38 nM T46781 D0J6AB 24748204 IC50 > 10 nM T46781 D0M0XB 10302451 IC50 > 10000 nM T46781 D0O0LS 25141092 IC50 > 1000 nM T46781 D0O6WV 24794418 IC50 = 78 nM T46781 D0P1CV 46191454 IC50 > 10000 nM T46781 D0Q7RE 16007391 IC50 = 0.3 nM T46781 D0Q9UX 16718576 IC50 = 4175 nM T46781 D0S4JK 24771867 IC50 = 1.5 nM T46781 D0S7HM 16041424 IC50 = 290 nM T46781 D0H7AC 51346455 IC50 = 5 nM T46781 C63WLY 89644 IC50 = 0.76 ug.mL-1 T46781 C5JE2Z 104860 IC50 = 0.98 ug.mL-1 T46781 CI1NA5 159926 IC50 = 0.65 ug.mL-1 T46781 CYBA43 177458 IC50 = 1.8 ug.mL-1 T46781 CN05AH 406563 IC50 = 1800 nM T46781 CB9F1O 447961 Ki = 57 nM T46781 C6A3LY 447962 Ki = 15 nM T46781 C1ZG2U 449087 IC50 > 10000 nM T46781 C76XNU 643953 IC50 > 3000 nM T46781 CQBY39 693946 IC50 = 7.665 nM T46781 C98SFI 698343 IC50 = 31 nM T46781 C8IAR2 5281657 IC50 = 3000 nM T46781 CI68PW 5283685 IC50 > 100000 nM T46781 CXK0S6 5283727 IC50 = 25100 nM T46781 C3BW1R 5327669 IC50 > 10000 nM T46781 CFW19M 5329009 IC50 = 7400 nM T46781 CDQ3M7 5359485 IC50 = 1 ug.mL-1 T46781 C54BYP 5360741 IC50 = 1.3 ug.mL-1 T46781 CDK3J0 5703619 IC50 = 2.3 nM T46781 C4G9WR 9547398 IC50 > 100000 nM T46781 C76CUP 9547698 IC50 > 100000 nM T46781 CTR6H5 9817349 IC50 = 1258.93 nM T46781 CBGE59 9833337 IC50 = 2900 nM T46781 C8BEZ2 9862708 IC50 > 10000 nM T46781 C2AYQ3 9924047 Ki = 207 nM T46781 CA05BZ 9925230 Ki = 575 nM T46781 CY0FT2 9946460 IC50 = 5070 nM T46781 CDT67L 9947412 Ki = 185 nM T46781 C1BX7I 9958417 Ki < 1 nM T46781 C75QCM 9969776 Ki > 1100 nM T46781 CVE1W8 10024433 Ki = 13 nM T46781 CR8DA1 10024683 IC50 > 100000 nM T46781 CLA93G 10047202 IC50 > 100000 nM T46781 C3LCH5 10047545 IC50 > 100000 nM T46781 CRQ01L 10094689 IC50 = 15 nM T46781 CKO01Z 10094732 IC50 = 14 nM T46781 CZV3U5 10111694 Ki > 1100 nM T46781 CV9B4X 10112611 Ki = 15 nM T46781 CD6GN4 10113529 Ki = 145 nM T46781 CCS0B9 10128386 Ki = 1 nM T46781 CLA2N6 10133600 Ki > 1100 nM T46781 CKL3V4 10134576 Ki > 40 nM T46781 C10WRQ 10153234 Ki < 1 nM T46781 CV73FD 10157920 Ki > 40 nM T46781 CQN8M3 10159519 Ki = 230 nM T46781 CY13QK 10175096 IC50 = 2 nM T46781 CR80BV 10175126 Ki = 1 nM T46781 CQ6J1C 10179215 Ki = 675 nM T46781 C3KHT0 10179373 Ki = 57 nM T46781 CXD4Z2 10180161 Ki = 51 nM T46781 CO08KZ 10182284 Ki = 250 nM T46781 CFUY91 10196758 Ki < 1 nM T46781 C7PEG0 10200408 Ki = 27 nM T46781 C1Z6EJ 10222721 Ki > 1100 nM T46781 C9FV7Z 10239608 Ki = 1 nM T46781 CZS9G0 10239769 Ki < 1 nM T46781 CSG14T 10239873 Ki < 1 nM T46781 C2PLB1 10239891 Ki < 1 nM T46781 C1KX3P 10248401 Ki = 9 nM T46781 CX7PD0 10252549 IC50 = 8 nM T46781 C28AEC 10268530 Ki = 590 nM T46781 CLQ3P2 10270356 Ki = 445 nM T46781 C13VMD 10273410 Ki = 83 nM T46781 C9V3SL 10289802 Ki < 1 nM T46781 CF9N7Y 10292186 Ki = 995 nM T46781 C8RD3V 10301884 IC50 = 8900 nM T46781 CNT46L 10311867 Ki = 1 nM T46781 CA23IN 10311891 Ki = 2 nM T46781 CD63MH 10312249 Ki < 1 nM T46781 C9J3RM 10320107 Ki = 9.7 nM T46781 CB45DL 10322308 IC50 = 25 nM T46781 CMY9D2 10340715 Ki = 6 nM T46781 CG2L4Z 10343860 IC50 = 20 nM T46781 CJ5W7O 10388447 IC50 = 18 nM T46781 CHLW70 10412796 IC50 = 9.5 nM T46781 C4CP7K 10423452 IC50 = 500 nM T46781 C7HBP6 10429593 IC50 > 10000 nM T46781 CC3L8Z 10430000 Ki = 9.4 nM T46781 C41GHN 10435854 Ki = 0.8 nM T46781 C83QWV 10714343 IC50 = 3890 nM T46781 C8G5WP 11210533 IC50 = 7290 nM T46781 C8T2NG 11211389 IC50 = 390 nM T46781 CQ4XT3 11224593 IC50 = 233 nM T46781 CK6U2S 11249084 IC50 = 135 nM T46781 CBOP58 11293798 Ki > 10000 nM T46781 C26BZX 11362471 Ki > 10000 nM T46781 CB45PJ 11362483 IC50 = 130 nM T46781 CWXB93 11397177 Ki > 10000 nM T46781 CT3VP7 11398307 IC50 = 45 nM T46781 CFJ6B2 11441375 IC50 = 118 nM T46781 CLZ3M8 11442557 IC50 = 48 nM T46781 C4Q7XD 11474276 IC50 = 220 nM T46781 C2Z7WP 11486459 IC50 = 46 nM T46781 C74BAE 11487958 IC50 = 99 nM T46781 C1UFM0 11497983 Ki = 0.37 nM T46781 CCVX84 11501979 IC50 > 100000 nM T46781 CR7MJ1 11508531 IC50 = 69000 nM T46781 CU4J8R 11523891 IC50 = 10 nM T46781 CCU8G9 11526006 IC50 = 2500 nM T46781 CL7X4Q 11530963 IC50 = 17000 nM T46781 CAWT72 11537541 IC50 > 100000 nM T46781 CTG83F 11539329 Ki > 6700 nM T46781 C6ZY9F 11545541 IC50 = 15000 nM T46781 C26ABY 11551547 IC50 = 15000 nM T46781 CZL4V1 11558640 IC50 = 3000 nM T46781 CACS26 11561968 Ki > 1000 nM T46781 CH05WP 11566279 IC50 = 700 nM T46781 CHR4Q6 11580435 IC50 = 260 nM T46781 C2CT6L 11587983 IC50 > 100000 nM T46781 CMIL86 11590363 Ki > 6700 nM T46781 CJ42AE 11603072 IC50 > 100000 nM T46781 C5ER3Q 11611230 IC50 = 34000 nM T46781 C5U4XY 11617275 IC50 > 100000 nM T46781 CUVW54 11617466 IC50 = 28000 nM T46781 CG6UC2 11624169 IC50 > 100000 nM T46781 CGX96V 11626927 IC50 > 5320 nM T46781 CIWA03 11632150 Ki = 2 nM T46781 CAN9R0 11632327 IC50 = 200 nM T46781 CL53BK 11639104 IC50 = 46000 nM T46781 C9T6SC 11640926 Ki > 6700 nM T46781 COF4I7 11645638 IC50 > 100000 nM T46781 CEV5X2 11646645 Ki = 4 nM T46781 C2CVI7 11647020 Ki = 6 nM T46781 CEBS68 11652621 IC50 > 100000 nM T46781 CKR96C 11653244 IC50 = 24000 nM T46781 C85HAQ 11655501 IC50 > 10000 nM T46781 CPNM76 11658909 IC50 = 17000 nM T46781 C8XGK5 11667761 IC50 > 100000 nM T46781 C8Z1YO 11681497 IC50 > 100000 nM T46781 CPQ19H 11681507 IC50 = 27000 nM T46781 CKC51F 11689306 IC50 = 34000 nM T46781 CU0E8O 11690457 Ki > 10000 nM T46781 CB0AP2 11705863 Ki > 1000 nM T46781 CFX9V2 11709165 IC50 = 34000 nM T46781 CH7DO8 11710518 IC50 > 50000 nM T46781 C8P3BC 11716968 IC50 = 12700 nM T46781 CW1VX7 11717761 IC50 = 930 nM T46781 C93KHF 11718021 Ki = 3 nM T46781 CJSV21 11744184 Ki = 18 nM T46781 CS5QL4 11749561 IC50 = 110 nM T46781 CV64JS 11750694 IC50 = 185 nM T46781 C9JT4S 11847343 IC50 = 45 nM T46781 CIR94K 11984538 IC50 = 431 nM T46781 CUDO23 11994441 IC50 = 630 nM T46781 C6H2RT 11994444 IC50 = 300 nM T46781 CN4JP1 11994445 IC50 = 1210 nM T46781 CM50UH 12000646 IC50 = 63 nM T46781 CGJ69E 12000661 IC50 = 31 nM T46781 CDGF78 15282555 IC50 = 500 nM T46781 C3YRU7 15295578 IC50 = 3200 nM T46781 CFPW41 16007116 Ki > 6700 nM T46781 CQR5O7 16042971 IC50 = 135 nM T46781 CW18IV 16070056 IC50 = 1640 nM T46781 CKR57M 16086104 IC50 > 25000 nM T46781 C16NRY 16086114 IC50 > 25000 nM T46781 C5VPH9 16129448 IC50 = 1370 nM T46781 C8FLH6 16202152 IC50 = 198 nM T46781 C6Q7FT 16221340 Ki = 510 nM T46781 C1BVO9 16221341 Ki < 1 nM T46781 CLX80H 16221342 Ki < 1 nM T46781 CIA5Y4 16221343 Ki < 1 nM T46781 CG9W2O 16221393 Ki < 1 nM T46781 CYJZ19 16221394 Ki < 1 nM T46781 CKT4N2 16719269 Ki = 23 nM T46781 C9IW5S 16730105 IC50 = 3000 nM T46781 CDVO81 16730408 IC50 = 46 nM T46781 CQ5H0C 16730410 IC50 = 130 nM T46781 C5D2NG 16730500 IC50 = 110 nM T46781 CPUN56 16730501 IC50 = 81 nM T46781 C38ZAH 16730583 IC50 = 810 nM T46781 CU5W8H 16730586 IC50 = 99 nM T46781 CTX68K 16730664 IC50 = 110 nM T46781 CMFL15 16730666 IC50 = 130 nM T46781 C23VWJ 16731303 IC50 = 62 nM T46781 C6S3YO 16731782 IC50 = 56 nM T46781 CK9CV4 16733534 IC50 = 77 nM T46781 CN0SA1 18450585 IC50 = 80 nM T46781 C7H4UM 18450846 IC50 = 13 nM T46781 CB9LG5 18451073 IC50 = 8 nM T46781 CSJ97R 18451176 IC50 = 11 nM T46781 CC9HG2 18451200 IC50 = 100 nM T46781 CQ1F3W 18451228 IC50 = 179 nM T46781 CW05LC 18451306 IC50 = 3280 nM T46781 CMQD24 18451374 IC50 = 487 nM T46781 CN42HV 18460835 IC50 = 1995.26 nM T46781 C5NCJ3 20604194 Ki = 153 nM T46781 CL81VC 21100709 IC50 = 735 nM T46781 C0KH4J 21106464 IC50 = 67000 nM T46781 CI4GS3 21106477 IC50 = 30000 nM T46781 CBL7W3 21106491 IC50 > 100000 nM T46781 C5W9CM 21106492 IC50 > 100000 nM T46781 CF59EQ 21106541 IC50 = 22000 nM T46781 C8IF5U 21991073 Ki = 120 nM T46781 C4V9UD 23545854 Ki = 115 nM T46781 CP01RM 23583059 IC50 = 26 nM T46781 CHM34D 23646072 IC50 = 1 nM T46781 CHU49V 24757938 IC50 = 18 nM T46781 C7YG1N 24759534 IC50 = 33 nM T46781 CQNP54 24764449 IC50 = 1000 nM T46781 CCPS81 24764502 IC50 > 35000 nM T46781 C2UOE0 24766030 IC50 > 50000 nM T46781 C74EZB 24815963 IC50 = 20 nM T46781 CEC8T9 24815964 IC50 = 3 nM T46781 C2EC0A 24815965 IC50 = 4.7 nM T46781 CIWJ29 24815966 IC50 = 3.6 nM T46781 C75MAH 24816055 IC50 = 1.7 nM T46781 CIC7O1 24816056 IC50 = 4.5 nM T46781 CO9Z0H 24822598 IC50 = 10 nM T46781 CA90EF 24822600 IC50 = 190 nM T46781 C4A6LB 24823090 IC50 = 62 nM T46781 CF6M3W 24823093 IC50 = 360 nM T46781 C0NLO8 24823094 IC50 = 680 nM T46781 C7D8PC 24823095 IC50 = 130 nM T46781 C14FLQ 24823250 IC50 = 16 nM T46781 C36BFD 24823252 IC50 = 385 nM T46781 C3GP7H 24880024 IC50 = 14 nM T46781 C43HWQ 24883287 IC50 > 10000 nM T46781 C8DA5Q 24883334 IC50 > 10000 nM T46781 C4V9GH 24894117 IC50 = 46000 nM T46781 CJH19T 24894883 IC50 = 9800 nM T46781 CJ14YB 24894884 IC50 = 4900 nM T46781 CB5TP8 24894992 IC50 = 43000 nM T46781 CP7QT2 24894995 IC50 = 2100 nM T46781 CFW40U 24894997 IC50 = 20000 nM T46781 CN13JF 24899915 IC50 = 0.22 ug.mL-1 T46781 CBWR97 24899916 IC50 = 1.1 ug.mL-1 T46781 C9F2JD 24899917 IC50 > 10 ug.mL-1 T46781 C64MTI 24900160 IC50 = 1.5 ug.mL-1 T46781 CO2I6Q 24900161 IC50 = 3 ug.mL-1 T46781 CT8OF0 24983254 IC50 = 134 nM T46781 CVF62Q 24983255 IC50 = 143 nM T46781 CX6FR3 24983298 IC50 = 454 nM T46781 CEQ1F2 24983299 IC50 = 47 nM T46781 CQ46VT 24983495 IC50 = 9 nM T46781 C4EG8R 24993189 IC50 > 10000 nM T46781 C3DI7Y 24995523 IC50 = 31 nM T46781 C2KY1G 25094210 IC50 <= 13 nM T46781 CR7X4M 25094243 IC50 = 24 nM T46781 CA6E0J 25094245 IC50 = 272 nM T46781 CC5NE0 25094283 IC50 = 129 nM T46781 CG3XC9 25124150 IC50 = 200 nM T46781 CO2IR5 25124816 IC50 = 4500 nM T46781 CH7EJ6 25138105 IC50 = 580 nM T46781 CVKD89 25138106 IC50 = 442 nM T46781 CWY2Q8 25138107 IC50 = 120 nM T46781 C8C2GV 25138109 IC50 = 54 nM T46781 C3KLX9 25138112 IC50 = 18 nM T46781 CX0RG8 25138115 IC50 = 13 nM T46781 C96IEQ 25138116 IC50 = 51 nM T46781 C8XW3Z 25138117 IC50 = 19 nM T46781 CZ07IH 25138118 IC50 = 61 nM T46781 C02EZG 25138119 IC50 = 22 nM T46781 C7LS2A 25138120 IC50 = 120 nM T46781 C80HOQ 25138349 IC50 = 59 nM T46781 CP6G0C 25143601 IC50 < 13 nM T46781 CGT1W6 25144294 IC50 < 13 nM T46781 C0CD4W 25144582 IC50 <= 13 nM T46781 CU7VR0 25144732 IC50 <= 13 nM T46781 CX5H1V 25145005 IC50 <= 13 nM T46781 CAO7K5 25145142 IC50 <= 13 nM T46781 CP3N2V 25145143 IC50 <= 13 nM T46781 C65YQG 25145144 IC50 <= 13 nM T46781 C6BWZ8 25145145 IC50 <= 13 nM T46781 C1VE8B 25145146 IC50 <= 13 nM T46781 CE31OI 25145147 IC50 <= 13 nM T46781 CORN76 25145280 IC50 <= 13 nM T46781 CF97LX 25145281 IC50 <= 13 nM T46781 CJ0ST3 25145282 IC50 <= 13 nM T46781 CFG67C 25145424 IC50 < 13 nM T46781 C52NQJ 25145568 IC50 < 13 nM T46781 C9N8UY 25145713 IC50 < 13 nM T46781 CX8LG5 25145714 IC50 < 13 nM T46781 C85ZKA 25145715 IC50 < 13 nM T46781 C78YWA 25145716 IC50 < 13 nM T46781 CL47VI 25145718 IC50 <= 13 nM T46781 CB21XV 25164469 Ki = 252 nM T46781 CNF0A8 25164674 Ki > 4900 nM T46781 CUX83H 25164675 Ki = 323 nM T46781 C1H7BF 25164677 Ki = 2366 nM T46781 CN50EI 25164678 Ki > 4900 nM T46781 C3XI7P 25164880 Ki > 4900 nM T46781 CX80QK 25164883 Ki > 4900 nM T46781 C6SD2A 25165081 Ki > 4900 nM T46781 C67TVH 25165085 Ki = 1577 nM T46781 C8J4KL 25165278 Ki = 26 nM T46781 CRJ6M7 25165279 Ki > 4900 nM T46781 C7RBX0 25165280 Ki > 4900 nM T46781 CPEY29 25165481 Ki > 4900 nM T46781 C70DRX 25165482 Ki > 4900 nM T46781 CE8D1W 25165860 Ki = 493 nM T46781 C6VZU2 25165861 Ki = 73 nM T46781 CVI70X 25166053 Ki = 15 nM T46781 C9VA1N 25166056 Ki = 16 nM T46781 C1JS9O 25166057 Ki = 42 nM T46781 CT94MS 25166059 Ki = 553 nM T46781 C5BM7F 25166250 Ki = 160 nM T46781 CCN25J 25166251 Ki = 186 nM T46781 CX8HY9 25166657 Ki = 66 nM T46781 C81WIV 25166867 Ki = 240 nM T46781 C9MR2O 25166869 Ki = 1800000 nM T46781 CAG1H6 25166870 Ki = 8666 nM T46781 CFE4O7 25166871 Ki = 2066 nM T46781 CGUC69 25167072 Ki = 5333 nM T46781 CF4G1L 25167074 Ki = 4340 nM T46781 C35ZXL 25167075 Ki = 834 nM T46781 C1CRJ7 25167076 Ki = 4450 nM T46781 C1IFX5 25167077 Ki = 3406 nM T46781 C2D3FP 25167078 Ki = 588 nM T46781 CP2W8I 25167079 Ki = 2125 nM T46781 CJO5A4 25167275 Ki = 810 nM T46781 C5KX0G 25167277 Ki > 4900 nM T46781 CQ5FJ8 25167278 Ki = 2805 nM T46781 C37YSX 25167280 Ki > 4900 nM T46781 CQ04LW 25171665 IC50 = 1840 nM T46781 CU9KV5 25171666 IC50 = 680 nM T46781 CN0I2H 25174496 IC50 = 28 nM T46781 COM37V 25174498 IC50 = 3 nM T46781 CQRJ38 25175157 IC50 = 172 nM T46781 CU4Z9Y 25175322 IC50 = 55 nM T46781 CCD92Y 25175326 IC50 = 938 nM T46781 CFX81M 25175327 IC50 = 525 nM T46781 CAN9J0 25175480 IC50 = 18 nM T46781 CJ76ZI 25175481 IC50 = 12 nM T46781 C2K3DU 25175482 IC50 = 4 nM T46781 C7TP4W 25175646 IC50 = 7 nM T46781 C7K9VO 25175648 IC50 = 41 nM T46781 CLG48V 25175948 IC50 = 127 nM T46781 CDK84B 25175951 IC50 = 82 nM T46781 CN9B1A 25176267 IC50 = 50 nM T46781 C5EQD8 25176269 IC50 = 12 nM T46781 CHMK36 25176588 IC50 = 480 nM T46781 CIB0V7 25176589 IC50 = 140 nM T46781 CLFM35 25206064 IC50 = 6000 nM T46781 C6FGQ1 25206346 IC50 = 4000 nM T46781 CNG96H 25210579 IC50 > 10000 nM T46781 CFL60D 25218594 IC50 = 5 nM T46781 CZW87R 25218595 IC50 = 1600 nM T46781 C1KR3Q 25218597 IC50 > 10000 nM T46781 C41TLH 42603880 IC50 = 69000 nM T46781 CRH7O2 42628076 IC50 = 1400 nM T46781 CM5QJ4 42628077 IC50 = 57 nM T46781 CU9E4P 42629114 IC50 > 10000 nM T46781 CO4FV0 42630578 IC50 = 1584.89 nM T46781 CJ5U1X 42639664 IC50 = 2.4 ug.mL-1 T46781 C1IYU0 44139710 IC50 = 55 nM T46781 C04IJO 44139711 IC50 = 1900 nM T46781 CN2G3C 44139712 IC50 = 3800 nM T46781 CTN41Y 44156909 IC50 = 3700 nM T46781 CN0X1C 44156917 IC50 > 10000 nM T46781 CLW80F 44160269 IC50 = 41000 nM T46781 C6CHK8 44177628 IC50 = 363 nM T46781 CD30LF 44177630 IC50 = 146 nM T46781 CCOE96 44177727 IC50 = 439 nM T46781 CT3G5K 44177728 IC50 = 1107 nM T46781 CGV40N 44177837 IC50 = 35 nM T46781 CTVZ96 44177838 IC50 = 175 nM T46781 C67ODN 44177840 IC50 = 41 nM T46781 CJE8L0 44177955 IC50 = 161 nM T46781 C7JY2E 44177956 IC50 = 155 nM T46781 CU08TA 44178067 EC50 = 285 nM T46781 CO1IM5 44178068 IC50 = 118 nM T46781 CO6HU7 44178069 IC50 <= 13 nM T46781 CX4R1O 44178070 IC50 <= 13 nM T46781 CNJ3Y1 44181654 IC50 = 11 nM T46781 CB0O2A 44186880 Ki > 4900 nM T46781 C9K7OP 44186882 Ki > 4900 nM T46781 CX0ZU8 44186885 Ki > 4900 nM T46781 CN8WB9 44189332 IC50 = 1 nM T46781 CNGV37 44189584 Ki > 4900 nM T46781 CK6I4N 44205288 IC50 = 2 nM T46781 CVH39F 44206601 IC50 = 13 nM T46781 CWM59J 44207068 IC50 = 1 nM T46781 CG1HI8 44207069 IC50 = 1 nM T46781 C6ZOR8 44207311 IC50 = 2 nM T46781 COAT76 44207312 IC50 = 0.8 nM T46781 CX1JE3 44207314 IC50 = 0.6 nM T46781 CAX3V9 44207547 IC50 = 1 nM T46781 CNA6M5 44207549 IC50 = 2 nM T46781 C1Q6YG 44208454 IC50 = 0.5 nM T46781 CK73NR 44219749 IC50 > 50000 nM T46781 CEL61X 44229839 IC50 > 10000 nM T46781 C1I9PA 44250391 IC50 = 23.7 nM T46781 CETQ79 44427518 IC50 = 8620 nM T46781 COPG94 44427519 IC50 > 50000 nM T46781 CLI16E 44465026 IC50 = 190 nM T46781 C9MV2P 44468256 IC50 = 53 nM T46781 CWG42F 44470318 IC50 = 66.3 nM T46781 CU4N2L 44518360 IC50 = 4 nM T46781 CA1VC7 44518362 IC50 = 24 nM T46781 C8YI9B 44518365 IC50 = 10 nM T46781 C7QU6G 44518503 IC50 = 1 nM T46781 C9GL6Y 44518504 IC50 = 0.9 nM T46781 CYH6P3 44520205 IC50 < 3 nM T46781 C4H0WR 44520206 IC50 = 36 nM T46781 CP56YC 44520407 IC50 = 38 nM T46781 CG37AY 44520577 IC50 = 33 nM T46781 C9HPB1 44520578 IC50 = 17 nM T46781 C94ZQD 44526805 IC50 = 67 nM T46781 C4WRN5 44541014 IC50 = 22200 nM T46781 C0LY6E 44552561 IC50 = 130 nM T46781 C7KRU3 44552562 IC50 = 162 nM T46781 C3VRO9 44557921 IC50 > 10000 nM T46781 CC7E4K 44564705 IC50 > 10000 nM T46781 C42ZEW 44564706 IC50 > 10000 nM T46781 C53MCK 44564747 IC50 = 1800 nM T46781 CDI31F 44564748 IC50 > 10000 nM T46781 CA17NT 44564749 IC50 > 10000 nM T46781 CMIZ20 44564750 IC50 > 10000 nM T46781 CSO9F8 44564751 IC50 > 10000 nM T46781 C8ATG9 44564787 IC50 = 7000 nM T46781 CM50GS 44564788 IC50 = 3100 nM T46781 C3Q0DX 44564789 IC50 > 10000 nM T46781 CP40XB 44564790 IC50 > 10000 nM T46781 C35NTB 44564791 IC50 > 10000 nM T46781 CJY83G 44564817 IC50 > 10000 nM T46781 CLK98G 44564818 IC50 > 10000 nM T46781 CF2D1K 44564819 IC50 > 10000 nM T46781 C3CQ9K 44564820 IC50 = 720 nM T46781 CI8V2L 44564821 IC50 > 10000 nM T46781 C9PO7J 44564860 IC50 > 10000 nM T46781 C16FJW 44564861 IC50 = 290 nM T46781 C8AMX5 44564862 IC50 = 750 nM T46781 CTR59U 44564863 IC50 > 10000 nM T46781 C9EY4C 44564864 IC50 > 10000 nM T46781 CG5Z7T 44564910 IC50 = 510 nM T46781 CU9O4C 44564911 IC50 > 10000 nM T46781 CXZ15S 44564954 IC50 > 10000 nM T46781 CZ78WJ 44564955 IC50 > 10000 nM T46781 CJ1X9V 44565013 IC50 = 2000 nM T46781 CN2Q3D 44565014 IC50 > 10000 nM T46781 CM2GN3 44565015 IC50 = 6400 nM T46781 C6RV9I 44565016 IC50 > 10000 nM T46781 CJC85A 44565069 IC50 = 920 nM T46781 CWFB42 44571820 IC50 = 1300 nM T46781 CCL85F 44575073 IC50 > 50000 nM T46781 CJX06P 44575126 IC50 = 8800 nM T46781 CE8FC7 44575127 IC50 = 10800 nM T46781 CAL46Y 44577971 IC50 = 22 nM T46781 C6RJZ5 44581565 IC50 = 23 nM T46781 CY6WV9 44591670 IC50 = 530 nM T46781 CG2RT4 44591671 IC50 = 57 nM T46781 C4MJZ5 44591672 IC50 = 42 nM T46781 CO2PF3 44591701 IC50 < 1 nM T46781 C28QLM 44605035 IC50 > 50000 nM T46781 C75XHS 44605037 IC50 = 45100 nM T46781 CU3RF1 45139989 IC50 > 10000 nM T46781 CQGZ06 45139991 IC50 > 10000 nM T46781 CRGD26 45266961 Ki = 49 nM T46781 CY15RC 45267893 Ki = 220 nM T46781 C9UX5Q 45269587 Ki = 59 nM T46781 CPO6K5 45271266 Ki = 105 nM T46781 C15MIZ 45272990 Ki = 52 nM T46781 CC95PQ 45375865 IC50 > 50000 nM T46781 CEOQ27 45375866 IC50 > 50000 nM T46781 C6OX0V 45375974 IC50 = 850 nM T46781 CX0HO6 45486156 IC50 = 270 nM T46781 C96BNW 46179972 IC50 = 2900 nM T46781 COL3S2 46182728 IC50 <= 13 nM T46781 CUA97D 46209401 IC50 = 66 nM T46781 C8ADR2 46214481 IC50 = 1995.26 nM T46781 CH0ZR1 46214482 IC50 = 12589.25 nM T46781 C2EZU8 46214649 IC50 = 7943.28 nM T46781 C5L1KH 46214650 IC50 > 10000 nM T46781 CRI6G5 46214652 IC50 = 10000 nM T46781 CRT51W 46214653 IC50 > 10000 nM T46781 CF57GK 46215462 IC50 = 100 nM T46781 CVW21C 46215644 IC50 = 3162.28 nM T46781 CZ58FY 46215814 IC50 = 3480 nM T46781 CO9H1K 46215816 IC50 = 1995.26 nM T46781 CT8G2A 46215988 IC50 = 25118.86 nM T46781 C28SJK 46215992 IC50 > 10000 nM T46781 C9JNT0 46216155 IC50 = 316.23 nM T46781 CD96WF 46216494 IC50 = 7943.28 nM T46781 CY3HW5 46224684 IC50 = 4300 nM T46781 C1U7IT 46225595 IC50 > 10000 nM T46781 C8YPN0 46225596 IC50 = 270 nM T46781 C34JTS 46225597 EC50 = 5000 nM T46781 CGD73B 46225598 IC50 = 520 nM T46781 C3E0PU 46225599 IC50 = 410 nM T46781 CRDY89 46225610 IC50 = 78 nM T46781 C0JMT8 46225611 IC50 = 48 nM T46781 CF0D5J 46225612 IC50 = 60 nM T46781 CFVO38 46225632 IC50 = 670 nM T46781 CLZ1O6 46225634 IC50 = 28 nM T46781 C07VDX 46225635 IC50 = 510 nM T46781 CT70DX 46225640 IC50 = 260 nM T46781 CJUF68 46225641 IC50 = 4800 nM T46781 C6AJ5N 46225647 IC50 = 41 nM T46781 C2WCV1 46225648 IC50 = 500 nM T46781 CBS96A 46225649 IC50 = 2100 nM T46781 C38BFC 46225657 IC50 = 300 nM T46781 CD0A6F 46225658 IC50 > 10000 nM T46781 C1B3KS 46225663 IC50 = 27 nM T46781 CU46XI 46225664 IC50 = 64 nM T46781 CO3HS2 46225665 IC50 = 62 nM T46781 C2UV1S 46225666 IC50 = 120 nM T46781 CX5B1G 46225667 IC50 = 90 nM T46781 C2Q9OH 46225668 IC50 = 8000 nM T46781 C16LEO 46225679 IC50 = 4200 nM T46781 CM14FH 46225680 IC50 = 800 nM T46781 CQS96E 46225681 IC50 = 1900 nM T46781 CJIK35 46225682 IC50 > 10000 nM T46781 C8S4QA 46225688 IC50 = 440 nM T46781 C7ON5A 46233287 IC50 > 10000 nM T46781 C1IZ5P 46236622 IC50 = 5 nM T46781 CW7F4D 46236768 IC50 = 8 nM T46781 CCSD82 46236769 IC50 = 5 nM T46781 CF2W4N 46237019 IC50 = 58 nM T46781 C97VFZ 46237140 IC50 = 46 nM T46781 CKTI63 46237141 IC50 = 276 nM T46781 CS35CW 46237142 IC50 = 24 nM T46781 CCZ65K 46237143 IC50 = 22 nM T46781 CGO1J5 46830766 Ki = 33 nM T46781 C2HJ1X 46830768 Ki = 3.8 nM T46781 C16JMS 46843255 IC50 = 83 nM T46781 CP1XL3 46846638 IC50 = 441 nM T46781 C17MQN 46846639 IC50 = 1870 nM T46781 CF6L2A 46846641 IC50 = 292 nM T46781 C5TJ2U 46846734 IC50 = 495 nM T46781 CB5Z6C 46846735 IC50 = 1720 nM T46781 CQWL17 46846948 IC50 = 402 nM T46781 C7NUY3 46847552 IC50 = 214 nM T46781 CCV16U 46847847 IC50 = 156 nM T46781 CC2O9R 46865656 IC50 = 15848.93 nM T46781 C8NB6R 46866505 IC50 = 9 nM T46781 CO3P0J 46866604 IC50 < 50000 nM T46781 CLS29B 46872626 IC50 > 10000 nM T46781 CJOM49 46880136 IC50 = 25500 nM T46781 CT48CR 46883054 IC50 = 420 nM T46781 C9ZVS1 46883055 IC50 = 620 nM T46781 C8NF4C 46883056 IC50 = 580 nM T46781 C2QBJ0 46883057 IC50 = 1400 nM T46781 CNO31X 46883058 IC50 > 10000 nM T46781 C3M8OQ 46883085 IC50 = 140 nM T46781 CMQ5F6 46883086 IC50 = 280 nM T46781 CXAD72 46883087 IC50 = 120 nM T46781 CS8CB4 46883134 IC50 = 2500 nM T46781 C5ETX6 46883135 IC50 = 6 nM T46781 CVG27D 46883136 IC50 = 8 nM T46781 CCQ6N9 46883137 IC50 = 21 nM T46781 C2U7OV 46883178 IC50 = 63 nM T46781 CI4VA7 46883179 IC50 = 600 nM T46781 CR48QI 46883180 IC50 = 5 nM T46781 C5EM0A 46883181 IC50 = 10 nM T46781 C5AYP7 46883321 IC50 = 5600 nM T46781 C5C9PR 46883322 IC50 > 10000 nM T46781 C7HPV1 46883323 IC50 = 1400 nM T46781 CRE96X 46885625 IC50 = 2 nM T46781 C75ZVX 46885628 IC50 = 6161 nM T46781 CZRY30 46885675 IC50 = 26 nM T46781 CK5WA6 46885676 IC50 = 104 nM T46781 CJBD40 46885677 IC50 = 169 nM T46781 C2O8RZ 46886323 IC50 = 660 nM T46781 CRAD15 46886342 IC50 = 47 nM T46781 CNJ50M 46886343 IC50 = 110 nM T46781 CP4O2N 46886344 IC50 = 46 nM T46781 CHL2F0 46886392 IC50 = 180 nM T46781 CKIH05 46886393 IC50 = 31 nM T46781 CMH09O 46886394 IC50 = 59 nM T46781 CQ6A0O 46886395 IC50 = 31 nM T46781 CT80IX 46888385 IC50 = 83 nM T46781 CEG84F 46888585 IC50 = 32 nM T46781 C38XJC 46888586 IC50 = 25 nM T46781 CE59WH 46888607 IC50 = 40 nM T46781 CE3N4O 46888608 IC50 = 50 nM T46781 CY48GN 46888609 IC50 = 16 nM T46781 CJ34VB 46888641 IC50 = 3 nM T46781 C4A9KL 46888642 IC50 = 1 nM T46781 CIG2O5 46888643 IC50 = 2 nM T46781 CA8X6N 46888676 IC50 = 64 nM T46781 CZN1S5 46888677 IC50 = 64 nM T46781 CYG5P0 46888678 IC50 = 85 nM T46781 CV6BH4 46888679 IC50 = 44 nM T46781 CDFP47 46888680 IC50 = 44 nM T46781 CB39WR 46888681 IC50 = 60 nM T46781 CHEB15 46888682 IC50 = 23 nM T46781 C7KM8F 46888683 IC50 = 26 nM T46781 C1SBV8 46888684 IC50 = 11 nM T46781 C2X3KJ 46888685 IC50 = 57 nM T46781 C53EWU 46888686 IC50 = 66 nM T46781 CW7C4L 46888746 IC50 = 1.4 nM T46781 C5RI8V 46888747 IC50 = 2.1 nM T46781 CXW80O 46888771 IC50 = 1.5 nM T46781 C0KN5S 46888772 IC50 = 5 nM T46781 CIN2Q6 46888773 IC50 = 4.7 nM T46781 C1O9ES 46888774 IC50 = 8.1 nM T46781 CX18GT 46889932 IC50 = 25 nM T46781 CM02UJ 46890253 IC50 = 100 nM T46781 CB7VI8 46890254 IC50 = 759 nM T46781 C7V3IA 46890314 IC50 = 55 nM T46781 CHE6A1 46890315 IC50 = 130 nM T46781 CTZ71Y 46898039 IC50 = 1.19 nM T46781 C5G2VE 46909588 IC50 > 5000 nM T46781 CL0O4U 46911726 Ki = 101 nM T46781 C28ELR 46912278 Ki = 63.1 nM T46781 CD4L7V 46912279 Ki = 79.43 nM T46781 C7S2HO 46913757 Ki = 316.23 nM T46781 CT46HI 46913758 Ki = 100 nM T46781 CVHG53 46913876 IC50 = 3154 nM T46781 CJ0M3S 46913877 IC50 = 310 nM T46781 CQLT07 46913878 IC50 = 235 nM T46781 C8Z1VS 46913879 IC50 = 356 nM T46781 CMVA69 46913880 IC50 = 312 nM T46781 CEC9O6 46914012 IC50 = 616 nM T46781 CJXV84 46916061 IC50 = 719 nM T46781 CS68OQ 46916062 IC50 = 906 nM T46781 CFE0B3 46916063 IC50 = 320 nM T46781 C60GAV 46929544 IC50 = 66 nM T46781 CF6D3X 46929545 IC50 > 25000 nM T46781 CZR46M 46929546 IC50 = 430 nM T46781 C50GPS 46929642 IC50 = 335 nM T46781 CZ4H0J 46929643 IC50 = 56 nM T46781 C20IBT 46929644 IC50 = 251 nM T46781 C3MTS0 46929645 IC50 = 542 nM T46781 C92GLN 46929646 EC50 = 89 nM T46781 C7QVB0 46929747 EC50 = 1450 nM T46781 CP34VL 46929748 EC50 = 15 nM T46781 CMF03G 46929749 EC50 = 28 nM T46781 CI93MV 46929750 EC50 = 20 nM T46781 C3IMQ5 46929751 EC50 = 15 nM T46781 CJ2E9Q 46929857 EC50 = 24 nM T46781 CV4X7L 49787166 IC50 = 1 nM T46781 C8FO0A 49800151 IC50 = 10540 nM T46781 CY3EO0 49800670 IC50 = 12 nM T46781 C8ML5D 49806794 IC50 = 294 nM T46781 C2XZ8A 49830351 IC50 = 50 nM T46781 CGOR85 49830358 IC50 = 16 nM T46781 CJ3SU6 49830359 IC50 = 9 nM T46781 CKO52Y 49830360 IC50 = 31 nM T46781 CF91RS 49843531 IC50 > 10000 nM T46781 C1BJ7D 49850390 IC50 = 61 nM T46781 C7JOA5 49850473 IC50 = 32 nM T46781 CA4QJ0 49867401 IC50 <= 13 nM T46781 CYKC34 50898605 IC50 = 367 nM T46781 CA06SB 50898682 IC50 = 289 nM T46781 CU2WV0 50898683 IC50 = 193 nM T46781 C6IHC3 50898684 IC50 = 278 nM T46781 C1FL0P 50898685 IC50 = 196 nM T46781 CP4CI5 50898686 IC50 = 783 nM T46781 CCS4B1 50898764 IC50 = 264 nM T46781 C5J2WG 50898765 IC50 = 318 nM T46781 C3MFH7 50898766 IC50 = 221 nM T46781 CU9K2Q 50898767 IC50 = 181 nM T46781 CX3J2C 50898768 IC50 = 176 nM T46781 CMG3J8 50898859 IC50 = 845 nM T46781 CRCT70 50909914 IC50 = 3162.28 nM T46781 C0XDI4 50909915 IC50 = 1000 nM T46781 CUJL92 50909916 IC50 = 158.49 nM T46781 C51DKX 50909917 IC50 = 1584.89 nM T46781 C2Y6QS 50938552 IC50 > 10000 nM T46781 C8IL9F 50994667 IC50 <= 13 nM T46781 C4QA8D 50994668 IC50 <= 13 nM T46781 CR0B8X 50994669 IC50 <= 13 nM T46781 C9UK6T 50994670 IC50 <= 13 nM T46781 CIF3W1 50994671 IC50 <= 13 nM T46781 CAZQ43 51003133 IC50 <= 13 nM T46781 C9NYP4 51036677 IC50 > 10000 nM T46781 C4WRY3 51037112 IC50 > 10000 nM T46781 CRI28Z 51037948 IC50 > 10000 nM T46781 CDU4Q5 51346827 Ki = 524 nM T46781 CYD4A2 51354035 IC50 = 1584.89 nM T46781 CW2T3N 51354036 IC50 = 5011.87 nM T46781 CH8NX6 51354037 IC50 = 1584.89 nM T46781 CK63DI 51354327 IC50 = 25.12 nM T46781 CC6PZ4 51354328 IC50 = 398.11 nM T46781 C2FVX4 51354329 IC50 = 50.12 nM T46781 CV06QD 51354330 IC50 = 316.23 nM T46781 CR3AC1 51354331 IC50 = 5011.87 nM T46781 CUXD62 51354613 IC50 = 199.53 nM T46781 C3G1VK 51354899 IC50 = 25118.86 nM T46781 CK7NP1 51354900 IC50 > 10000 nM T46781 CEDN75 51354901 IC50 = 5011.87 nM T46781 CB0EU1 51355190 IC50 = 1584.89 nM T46781 CYZ03E 51356852 IC50 = 7943.28 nM T46781 CL3S8F 51356853 IC50 = 12589.25 nM T46781 C67DUF 51356854 IC50 = 15848.93 nM T46781 CAU2F6 51356855 IC50 > 10000 nM T46781 CD07RV 51356856 IC50 > 10000 nM T46781 CFM5I7 51357137 IC50 = 7943.28 nM T46781 CP6R5J 51357138 IC50 = 25118.86 nM T46781 CWCJ29 51357417 IC50 = 1258.93 nM T46781 CS9WE1 51357418 IC50 = 3981.07 nM T46781 C5G7BY 51357419 IC50 > 10000 nM T46781 CBM4P9 51357696 IC50 = 1995.26 nM T46781 C65MXB 51357954 IC50 = 1000 nM T46781 CXA03W 52920796 IC50 <= 13 nM T46781 CG5IK8 52936268 IC50 = 579 nM T46781 C2UH4P 52940893 IC50 <= 13 nM T46781 CQB32I 52941003 IC50 <= 13 nM T46781 CC42PX 52942070 IC50 <= 13 nM T46781 C38PKY 52942116 IC50 <= 13 nM T46781 C31EGF 52942164 IC50 <= 13 nM T46781 CF1X3D 52942218 IC50 <= 13 nM T46781 C15XBH 52942244 IC50 <= 13 nM T46781 C7T8NP 52944489 IC50 <= 13 nM T46781 C5A1IX 52944643 IC50 <= 13 nM T46781 C93RQV 52944679 IC50 <= 13 nM T46781 C7EWH2 52945730 IC50 <= 13 nM T46781 C8MCU4 52945733 IC50 <= 13 nM T46781 C34WPX 52945791 IC50 <= 13 nM T46781 CIM9A5 52946956 IC50 <= 13 nM T46781 C0OAD7 52947107 IC50 <= 13 nM T46781 C0CJD8 52948167 IC50 <= 13 nM T46781 CRFY84 52948208 IC50 <= 13 nM T46781 CKSH24 52948244 IC50 <= 13 nM T46781 C8FMO5 52948247 IC50 = 50 nM T46781 CZ19SU 52948345 IC50 <= 13 nM T46781 CF8WT5 52949399 IC50 <= 13 nM T46781 C42QAS 52949563 IC50 <= 13 nM T46781 C4NAB3 53236443 IC50 = 1260 nM T46781 C2CT5J 53236670 IC50 = 260 nM T46781 C3M6LV 53236671 IC50 = 1140 nM T46781 C5YZB7 53236674 IC50 = 66 nM T46781 C5W0BJ 53236676 IC50 = 86 nM T46781 CZ5L6F 53239373 IC50 = 2230 nM T46781 C2WFI8 53239374 IC50 = 624 nM T46781 C0ZHF8 53239375 IC50 = 805 nM T46781 CD1EQ3 53239587 IC50 = 171 nM T46781 C1BGN8 53239589 IC50 = 136 nM T46781 C7XBV1 53239590 IC50 = 714 nM T46781 CD4M8I 53239593 IC50 = 112 nM T46781 CE8OY2 53317913 IC50 <= 13 nM T46781 CZS8K4 53319042 Ki > 4900 nM T46781 C24GBF 53319075 IC50 = 13 nM T46781 CUD21V 53320263 Ki = 1930 nM T46781 CEL08W 53320550 IC50 <= 13 nM T46781 CESA85 53323614 Ki > 4900 nM T46781 C64DPY 53339204 IC50 = 114 nM T46781 CJHT05 53339330 IC50 = 16 nM T46781 CK2WR9 53339442 IC50 = 44 nM T46781 C7FL6K 53339554 IC50 = 43.4 nM T46781 CD60WP 53339555 IC50 = 6.2 nM T46781 C5R3GK 53339557 IC50 = 15 nM T46781 CK1A5J 53339881 IC50 = 23 nM T46781 C09YVS 53339992 IC50 = 28 nM T46781 C0S2AT 53340111 IC50 = 23 nM T46781 C9FE3W 53340113 IC50 = 23 nM T46781 COE3J0 53340221 IC50 = 288 nM T46781 CC40ZF 53340223 IC50 = 27 nM T46781 CZ50GD 53340224 IC50 = 37.6 nM T46781 C56KAW 53340225 IC50 = 27.1 nM T46781 C8XD1E 53340226 IC50 = 169 nM T46781 C19MQP 53340227 IC50 = 13 nM T46781 C1HRW0 53340444 IC50 = 91 nM T46781 CN7GQ8 53340448 IC50 = 94.5 nM T46781 CY0K4W 53340450 IC50 = 10 nM T46781 CGK32Y 53340563 IC50 = 8.9 nM T46781 C3YXA8 53340567 IC50 = 63.2 nM T46781 CQ4ZE3 53340570 IC50 = 28.6 nM T46781 CP5G7E 53340685 IC50 = 293 nM T46781 CS1P2T 53340687 IC50 = 47 nM T46781 C2KO6F 53340688 IC50 = 11.9 nM T46781 C39HDM 53340809 IC50 = 146 nM T46781 C4PTV3 53340810 IC50 = 420 nM T46781 C1L9IC 53340811 IC50 = 850 nM T46781 CVG90B 53389651 IC50 > 10000 nM T46781 CZ1CI3 53469824 IC50 = 457 nM T46781 CXA92G 53484170 IC50 > 20000 nM T46781 C7UK2N 53484181 IC50 > 20000 nM T46781 CKD9H6 53484182 IC50 > 20000 nM T46781 CH05EO 53484183 IC50 > 20000 nM T46781 CAR45T 53484184 IC50 > 20000 nM T46781 CRN28X 54581311 IC50 = 251.19 nM T46781 CE1ZK6 54759168 IC50 > 10000 nM T46781 C9ZFS1 54764923 IC50 = 38100 nM T46781 CG76TH 56587958 IC50 = 193 nM T46781 C83VCG 56587966 IC50 = 42.9 nM T46781 C67EBW 56587967 IC50 = 226 nM T46781 CM8JX1 56604907 IC50 = 10000 nM T46781 C1ZA3C 56658055 IC50 = 28 nM T46781 CBO7D0 56658056 IC50 = 51 nM T46781 C8GJ9S 56658692 IC50 < 13 nM T46781 CK3A4Z 56658700 IC50 = 305 nM T46781 C1JD6Z 56658841 IC50 = 232 nM T46781 C98WRJ 56658842 IC50 = 128 nM T46781 CRTE61 56659304 IC50 = 6309.57 nM T46781 CQ82EC 56661565 IC50 = 6300 nM T46781 CA02LO 56661566 IC50 = 190 nM T46781 C7OMK2 56661568 IC50 = 637 nM T46781 CFXO67 56661569 IC50 = 49 nM T46781 C2Z9YO 56662177 IC50 = 194 nM T46781 CR50XZ 56662178 IC50 = 242 nM T46781 C8NGC7 56662179 IC50 = 2987 nM T46781 C3H0VQ 56662180 IC50 = 2501 nM T46781 CWM35E 56662181 IC50 > 20000 nM T46781 CB0VE5 56662182 IC50 > 20000 nM T46781 CXCY28 56662867 IC50 = 62 nM T46781 CC90EV 56662926 IC50 = 219 nM T46781 CEI39Q 56665634 IC50 = 2739 nM T46781 CG5K2Q 56665635 IC50 = 2517 nM T46781 CVEM27 56665636 IC50 > 20000 nM T46781 CDT3K4 56665637 IC50 > 20000 nM T46781 CCD3U6 56665765 IC50 = 143 nM T46781 C6B7WR 56666236 IC50 = 794.33 nM T46781 C45XIM 56666238 IC50 > 25118.86 nM T46781 CP4B3L 56666399 IC50 = 18 nM T46781 CK75JI 56666400 IC50 = 110 nM T46781 CO6N5S 56666401 IC50 = 33 nM T46781 C2JRW4 56666402 IC50 = 81 nM T46781 CA46RQ 56668419 IC50 = 179 nM T46781 CI5QR2 56668420 IC50 = 78 nM T46781 C9ZTL3 56669088 IC50 > 20000 nM T46781 CC8F0R 56669218 IC50 = 43 nM T46781 CXW95K 56669219 IC50 = 1227 nM T46781 C5OF9G 56669642 IC50 = 6309.57 nM T46781 C3C1XF 56669814 IC50 = 120 nM T46781 C9FR3E 56669815 IC50 = 252 nM T46781 CUP61N 56671791 IC50 = 398.11 nM T46781 CC0XQ2 56671934 IC50 = 420 nM T46781 C6TN3Z 56671935 IC50 = 58 nM T46781 C8R9TW 56672548 IC50 = 4588 nM T46781 C0ROQ7 56672549 IC50 = 8484 nM T46781 CI6K1R 56672550 IC50 > 20000 nM T46781 CC5NQ4 56672551 IC50 = 754 nM T46781 CY0PA7 56672679 IC50 = 84 nM T46781 C6E7WM 56673153 IC50 = 7943.28 nM T46781 C2Z1LP 56673154 IC50 = 1995.26 nM T46781 CHEK09 56673306 IC50 = 185 nM T46781 C59QTV 56675311 IC50 = 2490 nM T46781 C02ENW 56675312 IC50 = 15000 nM T46781 CJA2N4 56675924 IC50 = 2541 nM T46781 CWY32H 56676047 IC50 = 837 nM T46781 CN4US8 56676481 IC50 = 5011.87 nM T46781 C49LUC 56676482 IC50 = 12589.25 nM T46781 C2XE7T 56676636 IC50 > 3000 nM T46781 CP14LU 56678505 IC50 = 3162.28 nM T46781 C6RB1T 56678646 IC50 = 828 nM T46781 CCG1L8 56678647 IC50 = 1830 nM T46781 CO6EB7 56678649 IC50 = 1790 nM T46781 C2ZVP7 56678650 IC50 = 84 nM T46781 CF5YP1 56679374 IC50 < 13 nM T46781 CDS09F 56679795 IC50 = 1995.26 nM T46781 CU04BI 56679796 IC50 = 3981.07 nM T46781 CTEK36 56679797 IC50 = 1258.93 nM T46781 CO9P6E 56679965 IC50 = 110 nM T46781 C1GC5S 56679966 IC50 <= 13 nM T46781 CFVN60 56679967 IC50 = 26 nM T46781 CX3O6G 56681964 IC50 = 655 nM T46781 CWX2K6 56681967 IC50 = 29 nM T46781 C7ORA8 56681968 IC50 = 28 nM T46781 CAT9Y1 56681969 IC50 = 51 nM T46781 CLKP65 56682548 IC50 = 653 nM T46781 CW2YZ7 56682555 IC50 = 11000 nM T46781 C1JWN7 56682556 IC50 = 339 nM T46781 CS9YF2 56682557 IC50 > 20000 nM T46781 COM56E 56682674 IC50 = 561 nM T46781 C1KJD9 56683295 IC50 = 51 nM T46781 CAK91L 56955954 IC50 > 3600 nM T46781 C5YRF8 57328039 IC50 = 5 nM T46781 C03XBT 57328467 IC50 = 1580 nM T46781 CXJ35L 57328543 IC50 = 872 nM T46781 CCF61V 57328544 IC50 = 664 nM T46781 C39KXI 57328545 IC50 = 370 nM T46781 CP7UB8 57383477 IC50 = 11 nM T46781 C17KCM 57384256 IC50 = 6.3 nM T46781 CM61IS 57384257 EC50 = 3 nM T46781 CM3P5V 57384258 IC50 = 14.6 nM T46781 CVMQ60 57384259 IC50 = 293 nM T46781 CXS5L6 57384509 IC50 = 42.2 nM T46781 C8OL3E 57384510 EC50 = 3 nM T46781 CG7EX8 57384511 IC50 = 9.3 nM T46781 CWTD19 57384512 IC50 = 6.2 nM T46781 C08YUK 57384513 IC50 = 7 nM T46781 C0XIJ8 57387792 IC50 = 103 nM T46781 CSF58I 57387794 IC50 = 362 nM T46781 C7JO5P 57388019 IC50 = 44.8 nM T46781 C0B8GU 57388020 IC50 = 9 nM T46781 C4WE9B 57391179 IC50 < 0.2 nM T46781 CY10TP 57391180 IC50 > 10 nM T46781 C4CN6V 57396453 IC50 > 10 nM T46781 CU2PF5 57398440 IC50 = 97 nM T46781 C68VTP 57946373 IC50 = 17 nM T46781 C78UXM 57946415 IC50 = 199 nM T46781 CWL0A1 57946504 IC50 = 455.5 nM T46781 CI50KU 58167984 IC50 = 0.4 nM T46781 CL9P3V 58168008 IC50 = 1440 nM T46781 C87VTG 58168047 IC50 = 174 nM T46781 C6LQ3W 58168051 IC50 = 0.7 nM T46781 C6F3DH 58168083 IC50 = 79 nM T46781 CBU03C 58168094 IC50 = 6 nM T46781 CQK0L7 58168151 IC50 = 1 nM T46781 C3R6DT 58168169 IC50 = 1 nM T46781 CMR59F 58282865 IC50 < 13 nM T46781 C2I3QW 58486157 IC50 = 10 nM T46781 C7ZKF5 58486186 IC50 = 6.9 nM T46781 CBF7L4 58486208 IC50 = 13 nM T46781 CM91GS 58486210 IC50 = 7 nM T46781 CQPU86 58486223 IC50 = 8.5 nM T46781 C51FBH 58486335 IC50 = 2100 nM T46781 CL6Q5B 59503456 IC50 <= 13 nM T46781 CV7N4L 59503457 IC50 = 178 nM T46781 CT15SY 59503468 IC50 = 81 nM T46781 CN8A1T 59503488 IC50 = 282 nM T46781 C4TQG5 59503510 EC50 = 164 nM T46781 C6OP8J 59503511 IC50 > 3000 nM T46781 CK36AN 59503540 IC50 <= 13 nM T46781 CKSV12 59503547 IC50 <= 13 nM T46781 CE4C9L 59503584 IC50 = 193 nM T46781 CWB60P 59503611 IC50 = 28 nM T46781 CVLR79 59503615 IC50 = 70 nM T46781 CAC9V1 59503633 IC50 <= 13 nM T46781 CHPZ79 59503635 IC50 > 3000 nM T46781 CT47FC 59503644 IC50 <= 13 nM T46781 C1KYO9 59503657 IC50 = 261 nM T46781 CP9A8T 59503659 IC50 <= 13 nM T46781 C05AKO 59503686 IC50 = 30 nM T46781 C2MO0R 59503688 IC50 <= 13 nM T46781 CM3TJ8 59503701 IC50 = 44 nM T46781 CRM90T 59503709 EC50 = 327 nM T46781 C1MA6J 59503711 IC50 <= 13 nM T46781 C4P7KI 59503724 IC50 = 761 nM T46781 CY4VQ0 59503725 IC50 = 94 nM T46781 CHE68K 59503732 EC50 = 388 nM T46781 CX29EU 59503744 IC50 <= 13 nM T46781 C6CJU5 59503756 IC50 <= 13 nM T46781 C2SW7U 59503836 IC50 <= 13 nM T46781 CXJ63M 59603829 IC50 < 10 nM T46781 CQEU96 59603842 IC50 = 28 nM T46781 CRIW40 59825670 IC50 > 10000 nM T46781 C63REN 59825673 IC50 = 3 nM T46781 C3UW1D 59825681 IC50 = 7 nM T46781 CI4F9C 59825699 IC50 = 12 nM T46781 C9LWV7 59825704 IC50 = 6 nM T46781 CO34FC 59825742 IC50 = 2 nM T46781 C65BUA 59825756 IC50 = 11 nM T46781 C3ZSR4 59825772 IC50 = 10 nM T46781 CI8C9G 59825774 IC50 = 4 nM T46781 CZ8S5M 59825775 IC50 = 7 nM T46781 COH62U 60097413 IC50 > 5000 nM T46781 C1MR8Q 60097495 IC50 > 1000 nM T46781 CSZA16 60155724 IC50 > 3600 nM T46781 C4SGZ6 60165992 IC50 > 100000 nM T46781 C98NOD 60165993 IC50 > 100000 nM T46781 C3WIX5 60165994 IC50 > 100000 nM T46781 C0G5WC 60165995 IC50 > 100000 nM T46781 CEQ07N 60166135 IC50 > 100000 nM T46781 CRV13A 60166136 IC50 > 100000 nM T46781 CLP62H 60166137 IC50 = 62000 nM T46781 C9X0ZC 60166139 IC50 = 5500 nM T46781 CWPZ07 60166141 IC50 = 6000 nM T46781 C8ZJF7 66548458 IC50 > 100000 nM T46781 CGW4L5 66548650 IC50 > 100000 nM T46781 C7Q2CM 66548653 IC50 > 100000 nM T46781 CI41NJ 66548849 IC50 = 1700 nM T46781 CTJ64B 66548850 IC50 > 100000 nM T46781 CA42UL 66554658 IC50 = 398.11 nM T46781 CX25QN 66555696 IC50 = 50.12 nM T46781 CL0X8S 66555697 IC50 = 79.43 nM T46781 C2Y7FX 66555698 IC50 = 251.19 nM T46781 C8PST7 66556032 IC50 = 63.1 nM T46781 CV8JO4 66556033 IC50 = 158.49 nM T46781 CSZ6I5 66556035 IC50 = 100 nM T46781 C6SL1Q 66556036 IC50 = 630.96 nM T46781 CX6J3B 66556201 IC50 = 50.12 nM T46781 CHWG72 66556203 IC50 = 50.12 nM T46781 CVPT78 66556206 IC50 = 7943.28 nM T46781 C0F5HW 66556207 IC50 = 3981.07 nM T46781 C6E7CU 66556365 IC50 = 31.62 nM T46781 CR7JT9 66556366 IC50 = 100 nM T46781 CSM89V 66556371 IC50 = 316.23 nM T46781 CK9QI1 66556533 IC50 = 630.96 nM T46781 CA1Z4Q 66556534 IC50 = 2511.89 nM T46781 CNRZ13 66556535 IC50 = 398.11 nM T46781 C7MD5X 66556536 IC50 = 1258.93 nM T46781 C01RFU 66556542 IC50 = 630.96 nM T46781 CK0XR7 66560844 IC50 = 4 nM T46781 C79HET 66721774 IC50 = 18 nM T46781 C6A3TN 66759619 IC50 > 20000 nM T46781 CY36UH 66760355 IC50 = 6500 nM T46781 CE20FQ 66760840 IC50 = 160 nM T46781 CZ5JA1 66761050 IC50 = 17400 nM T46781 CP94KX 66761096 IC50 = 3000 nM T46781 CLQ51N 66761102 IC50 > 20000 nM T46781 CE49GC 67098566 Ki = 10 nM T46781 CT35MO 67127525 IC50 = 44 nM T46781 C0CL1R 67127737 IC50 = 135 nM T46781 C37NKO 67129970 IC50 > 10000 nM T46781 CK80LJ 67130050 IC50 > 10000 nM T46781 CV63UL 67240318 IC50 > 10000 nM T46781 CUI07E 67378360 IC50 = 16 nM T46781 C6D3QJ 67448476 IC50 = 6.9 nM T46781 C7N4ZS 68034365 IC50 = 9400 nM T46781 C32TVX 68230798 IC50 = 2400 nM T46781 C4M9LX 68289700 IC50 = 63.1 nM T46781 C07JAL 68290083 IC50 = 1995.26 nM T46781 CC70KY 68290508 IC50 = 1995.26 nM T46781 CUR2V0 68290592 IC50 > 100000 nM T46781 C7U4VX 68290829 IC50 = 4500 nM T46781 C24IRX 68290838 IC50 > 100000 nM T46781 CY60FW 68290875 IC50 > 100000 nM T46781 C7GK8I 68290918 IC50 > 100000 nM T46781 CC8IR2 68290919 IC50 > 100000 nM T46781 CVB70Q 68291007 IC50 = 2300 nM T46781 C0OIP9 68291028 IC50 > 100000 nM T46781 C7CZX6 68291099 IC50 > 100000 nM T46781 CEZI21 68291184 IC50 = 34000 nM T46781 C8CSV6 68291375 IC50 > 100000 nM T46781 C2S0CH 68291448 IC50 > 100000 nM T46781 CIB52Q 68309298 IC50 = 501.19 nM T46781 CBGL83 68309299 IC50 = 251.19 nM T46781 CWDS89 68310172 IC50 = 501.19 nM T46781 CM5J8Z 68649048 IC50 = 1 nM T46781 CYI75G 68678653 IC50 = 27.3 nM T46781 C7GRV2 68755406 IC50 > 10000 nM T46781 C8WZE0 68777669 IC50 = 118 nM T46781 COK9X0 68779704 IC50 = 43 nM T46781 C47JKD 68780376 IC50 = 197 nM T46781 CC42HY 68780543 IC50 = 99 nM T46781 CZ2F5K 68780558 IC50 = 32 nM T46781 CWQP24 68780634 IC50 = 29 nM T46781 C71UOK 68780741 IC50 = 12 nM T46781 C6LY1M 68781121 IC50 = 28 nM T46781 C0G1NM 68781294 IC50 = 31 nM T46781 C62GYI 68781318 IC50 = 252 nM T46781 C60FTP 68781521 IC50 = 15 nM T46781 CJBW54 68781929 IC50 = 25 nM T46781 C8KP2A 68782417 IC50 = 8 nM T46781 CNEM15 68782426 IC50 = 19 nM T46781 CP5IF4 68782618 IC50 = 45 nM T46781 C5W7QY 68782756 IC50 = 26 nM T46781 C49PZJ 68782797 IC50 = 15 nM T46781 C8W5RV 68782804 IC50 = 12 nM T46781 CE84YM 68782852 IC50 = 145 nM T46781 CVML10 68783198 IC50 = 27 nM T46781 C76VIM 68783233 IC50 = 51 nM T46781 CE0YK8 68783378 IC50 = 29 nM T46781 CYE91N 68783396 IC50 = 12 nM T46781 C0Q4XO 68783521 IC50 = 8 nM T46781 C0HA8V 68783839 IC50 = 42 nM T46781 C5DGR9 69036886 IC50 = 163 nM T46781 C3GTU1 69762142 IC50 > 10000 nM T46781 C2AZ4X 69787126 IC50 = 39.81 nM T46781 CZ4OY5 70681030 IC50 = 16 nM T46781 CPOV92 70681032 IC50 = 4 nM T46781 COHI26 70681033 IC50 = 13 nM T46781 C3NVZ6 70681070 IC50 = 50 nM T46781 C56ZER 70681071 IC50 = 6 nM T46781 CH6S7Q 70681377 IC50 = 1 nM T46781 CV24XU 70681532 IC50 = 18 nM T46781 CRYW49 70681533 IC50 = 60 nM T46781 C7EH1D 70683155 IC50 = 81 nM T46781 C1R6HY 70683192 IC50 = 5 nM T46781 CJMQ50 70683427 IC50 <= 13 nM T46781 CRE52C 70683471 IC50 = 529 nM T46781 CFN46P 70683472 IC50 = 11 nM T46781 CRA3I8 70683473 IC50 = 2 nM T46781 CXTS83 70683500 IC50 = 70 nM T46781 C81YOT 70683501 IC50 = 52 nM T46781 CDB0H6 70683503 IC50 = 21 nM T46781 C3NCF2 70683641 IC50 = 4 nM T46781 CY51SV 70683642 IC50 = 5 nM T46781 CD29LB 70684383 IC50 > 12500 nM T46781 C0XPO9 70684384 IC50 = 36 nM T46781 CRK92N 70685231 IC50 = 30 nM T46781 CID9O3 70685233 IC50 = 478 nM T46781 C6QZ5U 70685271 IC50 = 4 nM T46781 CPTG79 70685272 IC50 = 4 nM T46781 C7NP5X 70685550 IC50 = 45 nM T46781 CVFU50 70685579 IC50 = 5 nM T46781 C39GML 70685599 IC50 = 114 nM T46781 C4PW8O 70685778 IC50 = 30 nM T46781 CN3E5T 70685779 IC50 = 4 nM T46781 CA0FE8 70687386 IC50 = 43 nM T46781 CQH9A0 70687387 IC50 = 24 nM T46781 CMA7J1 70687388 IC50 = 7 nM T46781 C6DAJ0 70687420 IC50 = 12 nM T46781 C6FO8B 70687421 IC50 = 5 nM T46781 CZEN15 70688644 IC50 > 12500 nM T46781 CEGM27 70689447 IC50 = 29 nM T46781 C80CWD 70689448 IC50 = 93 nM T46781 C01WIM 70689476 IC50 = 4 nM T46781 CH30CI 70689776 IC50 = 177 nM T46781 C1CJ8S 70689777 IC50 = 8 nM T46781 CCD49V 70689801 IC50 = 6 nM T46781 CAE31H 70689940 IC50 = 4 nM T46781 C1IN7G 70689941 IC50 = 4 nM T46781 CI27NT 70690992 IC50 = 66 nM T46781 CN15SY 70691556 IC50 = 38 nM T46781 CS1G5L 70691585 IC50 = 38 nM T46781 CDWB98 70691595 IC50 = 5 nM T46781 C5MT8A 70691596 IC50 = 4 nM T46781 CC5A4K 70692098 IC50 = 4 nM T46781 CADI76 70692099 IC50 = 40 nM T46781 CW9MY1 70693675 IC50 = 19 nM T46781 C2L6OP 70693678 IC50 = 22 nM T46781 CNRC67 70693679 IC50 = 4 nM T46781 CJZ5E1 70693680 IC50 = 36 nM T46781 C2ZIB3 70693989 IC50 = 68 nM T46781 CA4DU8 70693990 IC50 = 18 nM T46781 C05FGA 70693991 IC50 = 17 nM T46781 C4IV6B 70693993 IC50 <= 13 nM T46781 CWM0K6 70695185 IC50 = 16 nM T46781 CL71AV 70695758 IC50 = 31 nM T46781 C2EI9Z 70695759 IC50 = 25 nM T46781 CZ4W6K 70695760 IC50 = 733 nM T46781 C2QJ8X 70695789 IC50 = 18 nM T46781 CPW57H 70695790 IC50 = 23 nM T46781 CC8WG5 70695791 IC50 = 4 nM T46781 C2UMZ0 70695792 IC50 = 40 nM T46781 C1SX4Q 70695793 IC50 = 3 nM T46781 CA6HC7 70696091 IC50 = 23 nM T46781 CQIS80 70696112 IC50 = 66 nM T46781 CW5Z7B 70696113 IC50 = 8 nM T46781 C1U7FS 70696114 IC50 = 48 nM T46781 C76JFM 70696269 IC50 = 1000 nM T46781 CNI64Y 70696270 IC50 = 4 nM T46781 CHAY50 70696941 IC50 = 450 nM T46781 C5RY7I 70702144 IC50 = 50.2 nM T46781 CVX3W4 70702148 IC50 = 1000 nM T46781 CGV53S 70702149 IC50 = 93.9 nM T46781 C3CT2W 70702150 IC50 = 123 nM T46781 CQI41A 70702151 IC50 = 180 nM T46781 C2T0RP 70702152 IC50 = 174 nM T46781 C0Q5XG 70702153 IC50 = 361 nM T46781 CVNR83 70702154 IC50 = 1510 nM T46781 C4F2HG 70702155 IC50 < 1000 nM T46781 CZ19MK 70702156 IC50 < 1000 nM T46781 CR50CX 70702157 IC50 < 1000 nM T46781 CB5Z1F 70702158 IC50 = 30 nM T46781 CZ19LH 70702159 IC50 < 1000 nM T46781 CL5P4C 70702160 IC50 < 1000 nM T46781 CXY46F 70702161 IC50 = 56.6 nM T46781 CQK2G1 70702162 IC50 = 83.7 nM T46781 CY2P3B 70702164 IC50 = 106 nM T46781 COM14R 71044759 IC50 < 13 nM T46781 CFTP07 71044863 IC50 < 13 nM T46781 CZ29NF 71113911 IC50 = 100 nM T46781 CT1L2V 71113915 IC50 = 79.43 nM T46781 CKOE90 71451677 IC50 = 58 nM T46781 CEBO91 71452977 IC50 = 500 nM T46781 C47GYB 71454279 IC50 = 148 nM T46781 CCN01X 71547862 IC50 > 10000 nM T46781 CB3SO2 71567006 IC50 > 10000 nM T46781 CDJY72 71568837 IC50 = 5100 nM T46781 CRX81Q 71575642 IC50 > 10000 nM T46781 CZ31PU 71583657 IC50 > 10000 nM T46781 CCXT12 71614919 IC50 = 21 nM T46781 CS62NH 71698376 IC50 = 1711 nM T46781 CI8X1R 71698379 IC50 = 985.2 nM T46781 C60BIX 71763463 IC50 = 25.5 nM T46781 CMLF37 71814652 IC50 > 10000 nM T46781 CPNQ29 71814653 IC50 = 6900 nM T46781 CY21KG 71814654 IC50 = 1700 nM T46781 CJ98FV 71814655 IC50 = 1500 nM T46781 C9GS6R 71814656 IC50 = 1700 nM T46781 CKZ5W3 71815103 IC50 = 10.5 nM T46781 CCV20F 71815104 IC50 = 16.4 nM T46781 C4Q6FE 71815105 IC50 = 25 nM T46781 CJ9OX6 71815106 IC50 = 29.6 nM T46781 CZY84B 71815389 IC50 = 87.4 nM T46781 C2R4SM 71815390 IC50 = 791.1 nM T46781 CT0A1Y 71815452 IC50 = 209.4 nM T46781 CSA3K0 71815640 IC50 = 14.9 nM T46781 CK69NO 71815643 IC50 = 127.6 nM T46781 CGV20M 71815692 IC50 > 1000 nM T46781 C9HTL7 71815698 IC50 = 102.2 nM T46781 C8X3RA 71815744 IC50 = 55.5 nM T46781 CUQK27 71815745 IC50 > 1000 nM T46781 C38MPZ 71815746 IC50 = 1.8 nM T46781 C2XCQ0 71815749 IC50 = 10.7 nM T46781 C3Z9XP 71815811 IC50 = 6.5 nM T46781 COP37R 71815812 IC50 = 5.3 nM T46781 CZHF40 71815813 IC50 = 7.7 nM T46781 CUP32D 71815814 IC50 = 15 nM T46781 CAU21X 71815815 IC50 = 40.9 nM T46781 CC1Q2L 71815881 IC50 = 29.8 nM T46781 C6NV5E 71815882 IC50 = 18.4 nM T46781 CC1T4S 71815884 IC50 = 158.7 nM T46781 CWOS79 71815948 IC50 = 1.2 nM T46781 CO6EQ1 71815949 IC50 = 3 nM T46781 CBF15Z 71816016 IC50 = 3 nM T46781 C3ZX5P 71816017 IC50 = 2.3 nM T46781 CG01VI 71816018 IC50 > 1000 nM T46781 CCM0E5 71816019 IC50 = 1.5 nM T46781 CWUH04 71816084 IC50 = 30.6 nM T46781 CY8CM3 71816085 IC50 = 16.8 nM T46781 C3VT2G 71816086 IC50 = 217.9 nM T46781 CD28XR 71816087 IC50 = 0.4 nM T46781 CPU41Q 71816088 IC50 = 7.6 nM T46781 CE04IC 71816173 IC50 = 7 nM T46781 CI8P1V 71816174 IC50 = 80 nM T46781 C5SVI9 72194531 IC50 = 50 nM T46781 CL6PC8 72194532 IC50 = 91.7 nM T46781 CFTK59 72705466 Ki = 19952.62 nM T46781 C1CU0H 72705467 Ki = 630.96 nM T46781 CX2AW3 72705468 Ki = 79.43 nM T46781 CVK4Z3 72705469 Ki = 5011.87 nM T46781 C4ND6R 72705470 Ki = 5.012 nM T46781 CT67YO 72706106 Ki > 19952.62 nM T46781 CA6ZB2 72734882 IC50 = 17 nM T46781 CG3E2H 72734883 IC50 = 9 nM T46781 COQC81 72734884 IC50 = 169 nM T46781 C8BW7J 72734885 IC50 = 18600 nM T46781 CA58QS 72734886 IC50 = 24650 nM T46781 CCP73J 72735062 IC50 = 693 nM T46781 CHJ1P0 72735063 IC50 = 3447 nM T46781 CMD43O 72735064 IC50 = 1676 nM T46781 CJ4L9T 72735065 IC50 = 3910 nM T46781 CID56Z 72735066 IC50 = 1817 nM T46781 C5P8ZH 72735248 IC50 = 3045 nM T46781 CFR12B 72737418 IC50 = 441 nM T46781 CRK95J 72737419 IC50 = 7095 nM T46781 C4CT0M 72737420 IC50 = 97 nM T46781 C2T1BW 72737421 IC50 = 1087 nM T46781 CQ3O1Z 72737597 IC50 = 2 nM T46781 CA62KV 72737598 IC50 = 8 nM T46781 C4FY5U 73346554 Ki = 251.19 nM T46781 CPGD07 73348027 Ki > 19952.62 nM T46781 C05XEV 73348028 Ki > 19952.62 nM T46781 CUW70Y 73348034 Ki = 316.23 nM T46781 CFEU95 73348035 Ki = 79.43 nM T46781 C6K0UL 73348036 Ki = 3162.28 nM T46781 CD6KE7 73349574 Ki = 0.5012 nM T46781 CV8UR4 73351136 Ki = 251.19 nM T46781 CAS60G 73352600 Ki = 501.19 nM T46781 CX75YR 73352604 Ki = 398.11 nM T46781 C5YKB4 73352605 Ki = 316.23 nM T46781 C03YUP 73355623 Ki = 2511.89 nM T46781 C1A9PR 73357167 Ki = 398.11 nM T46781 C3UC9H 73891099 IC50 = 2510 nM T46781 CV8QX0 76310169 IC50 = 22600 nM T46781 C42MXW 76310923 IC50 = 889 nM T46781 C0MR6F 76310924 IC50 = 1680 nM T46781 C81ECP 76313984 IC50 > 100000 nM T46781 C7HYN3 76313985 IC50 > 100000 nM T46781 C9MG7U 76314564 IC50 = 18800 nM T46781 CRLG27 76317532 IC50 > 100000 nM T46781 CU8EW0 76318141 IC50 = 156 nM T46781 C80VJZ 76318142 IC50 = 1380 nM T46781 C6ZOM5 76321826 IC50 = 5920 nM T46781 C5MRE6 76321827 IC50 = 2300 nM T46781 CA5L4W 76324771 IC50 = 20600 nM T46781 CH8Q9D 76324874 IC50 = 47000 nM T46781 C8Z6XR 76325460 IC50 = 299 nM T46781 CKZ4F9 76325461 IC50 = 1300 nM T46781 CTA86L 76325462 IC50 = 2820 nM T46781 C9GO0P 76328313 IC50 = 8690 nM T46781 CN15WO 76328435 IC50 = 16000 nM T46781 CT1R6E 76329005 IC50 = 284 nM T46781 CT4FE5 76329006 IC50 = 12100 nM T46781 C39FTZ 76335685 IC50 > 100000 nM T46781 CS0CN8 76335739 IC50 > 100000 nM T46781 C0PRE8 76336290 IC50 = 2470 nM T46781 CF1JW0 76336291 IC50 = 1440 nM T46781 CQ2SU8 78673832 IC50 = 689 nM T46781 CE0W9R 78673833 IC50 = 23100 nM T46781 CK61HY 85469442 IC50 > 10000 nM T46781 CV8UZ1 86278565 IC50 = 4030 nM T46781 C1HW4B 89735655 IC50 = 4600 nM T46781 C9YWN1 89790691 IC50 = 290 nM T46781 C61TVX 89857999 IC50 = 6.5 nM T46781 CQW14S 89858004 IC50 = 1.5 nM T46781 CA4F0J 89858007 IC50 = 1.3 nM T46781 CU85OG 89858012 IC50 = 209.3 nM T46781 C76NRF 89858053 IC50 = 14.3 nM T46781 CF17VX 89858058 IC50 = 18.4 nM T46781 C3BHE0 89858077 IC50 = 250.6 nM T46781 C2ECL1 89858082 IC50 = 1.9 nM T46781 CGC5Z7 89858094 IC50 = 32.5 nM T46781 CM4WJ2 89868555 IC50 = 347 nM T46781 CN76VK 89912923 IC50 = 158.49 nM T46781 CV64KY 90183363 IC50 > 10000 nM T46781 CL4JO2 90183809 IC50 = 6190 nM T46781 C28WQY 90431726 IC50 = 4.2 nM T46781 CY0UC4 90645194 IC50 > 10000 nM T46781 C0Y8ZK 91933875 IC50 > 1000 nM T46781 C9BL4M 92045136 IC50 = 132 nM T46781 CS2J0P 101879051 IC50 = 2205 nM T46781 C0R2OH 101879052 IC50 = 587 nM T46781 CRI0S4 101891768 IC50 > 10000 nM T46781 CXS96K 101902488 IC50 = 5940 nM T46781 CGB54P 101902999 IC50 = 720 nM T46781 CG62HP 101903000 IC50 = 480 nM T46781 CT3P6B 102156535 IC50 = 1800 nM T46781 C5N1VZ 102581295 IC50 > 10000 nM T46781 CICU38 118213763 IC50 = 7 nM T46781 CS5C8W 118684133 IC50 = 4.6 nM T46781 CRS34C 118705500 IC50 > 100000 nM T46781 CY7BI2 118706214 IC50 > 10000 nM T46781 C2IN3C 118710236 IC50 = 5.9 nM T46781 CF2YR1 118710237 IC50 = 93 nM T46781 CS9VP0 118710238 IC50 = 252.6 nM T46781 CE13CO 118710415 IC50 = 47500 nM T46781 CFJ1N6 118710418 IC50 = 13800 nM T46781 C6O7DN 118710473 IC50 = 31900 nM T46781 CUZL50 118710481 IC50 = 21800 nM T46781 CX0W3J 118710482 IC50 = 63200 nM T46781 CX58DI 118716791 IC50 = 155 nM T46781 CD9X2B 118716796 IC50 = 5910 nM T46781 C2YJ0O 118716797 IC50 > 30000 nM T46781 CL3UO9 118716798 IC50 > 30000 nM T46781 C71BAM 118716799 IC50 > 30000 nM T46781 CU4EL6 118716806 IC50 = 14300 nM T46781 C7XE9K 118716988 IC50 = 172 nM T46781 CS8Q2C 118716989 IC50 = 292 nM T46781 CI5W9H 118720010 IC50 > 10000 nM T46781 COQ9S4 118720011 IC50 > 10000 nM T46781 C3KLI5 118723185 IC50 > 100000 nM T46781 C9XNG5 118724918 IC50 = 21.5 nM T46781 CG25JP 118725515 IC50 = 5 nM T46781 C6XW9J 118725516 IC50 = 127 nM T46781 CJQE38 118725517 IC50 = 2 nM T46781 CS1FU0 118725519 IC50 = 6 nM T46781 C3QD8O 118725520 IC50 = 7 nM T46781 C6LWF1 118725521 IC50 = 8 nM T46781 CO30HX 118725522 IC50 = 25 nM T46781 CDP96A 118725523 IC50 = 6 nM T46781 CR95GT 118725524 IC50 = 4 nM T46781 C3OP2A 118725526 IC50 = 2 nM T46781 CT8Z0C 118725528 IC50 = 5 nM T46781 CAK4Y3 118725529 IC50 = 3 nM T46781 C46DME 118725530 IC50 = 26 nM T46781 C8I6GM 118725531 IC50 = 8 nM T46781 CG3JU9 118725532 IC50 = 180 nM T46781 CGB27X 118725533 IC50 = 2 nM T46781 CVTN86 118725534 IC50 = 7 nM T46781 C6ML4Z 118725535 IC50 = 1100 nM T46781 CT7U4L 118734734 IC50 = 430 nM T46781 CYO74T 118734736 IC50 = 395 nM T46781 C94KIG 122184152 IC50 = 3300 nM T46781 C0SLH3 122184153 IC50 = 8200 nM T46781 C9ATR0 122184169 IC50 = 2500 nM T46781 C5AFZ6 122191639 IC50 = 110 nM T46781 C4X7SD 122192466 IC50 > 10000 nM T46781 C18FWG 122197326 IC50 = 573 nM T46781 C8CMZ9 122197327 IC50 = 621 nM T46781 CSP09Z 122197328 IC50 = 197 nM T46781 CYX60U 122197329 IC50 = 232 nM T46781 CE5C3B 122197330 IC50 = 387 nM T46781 C1VGJ2 122197331 IC50 = 589 nM T46781 CBYC49 126617676 IC50 = 114.4 nM T46781 C50QVG 127027240 IC50 = 49500 nM T46781 CHN0C6 127028483 IC50 = 10200 nM T46781 CLQE43 127028484 IC50 = 20100 nM T46781 C26ZFL 127028485 IC50 = 364 nM T46781 CDT31P 127029393 IC50 = 16300 nM T46781 CA4UH3 127029997 IC50 = 36500 nM T46781 C4W7TU 127031218 IC50 = 32100 nM T46781 C0PUM7 127031807 IC50 = 2190 nM T46781 CTB34H 127031808 IC50 = 54800 nM T46781 CZ02HG 127031810 IC50 = 40700 nM T46781 CR18NB 127032078 IC50 = 15200 nM T46781 C4JF8H 127040661 IC50 = 16 nM T46781 C7P5MY 127040994 IC50 = 157 nM T46781 CL0I6O 127044234 IC50 = 10200 nM T46781 CJT4C2 127044236 IC50 = 600 nM T46781 CTO95Y 127044392 IC50 = 700 nM T46781 CJCQ76 127044457 IC50 = 50400 nM T46781 CBHG81 127044600 IC50 = 49400 nM T46781 CA6ES3 127053398 IC50 = 1330 nM T46781 CRJ04D 127053399 IC50 = 7300 nM T46781 CO8Z2N 129900111 EC50 = 11 nM T46781 C0FM1R 130196825 IC50 = 8580 nM T46781 CL26YS 132005219 IC50 = 80 nM T46781 CP32GB 132005220 IC50 = 290 nM T46781 CUN18W 132005225 IC50 = 150 nM T46781 CD84OI 132005228 IC50 = 120 nM T46781 C9VDI0 132005229 IC50 = 16 nM T46781 C7ASP9 132005246 IC50 = 120 nM T46781 C5W9LN 132005323 IC50 = 630 nM T46781 CQ6GO2 132005326 IC50 = 130 nM T46781 C1MCE8 134136983 IC50 = 31 nM T46781 CI8Y4X 134139821 IC50 = 64 nM T46781 CE7Q4G 134140427 IC50 > 25000 nM T46781 CX5C8B 134140540 IC50 = 49 nM T46781 CWB68E 134143937 IC50 > 1000 nM T46781 CQJM72 134144731 IC50 = 26 nM T46781 CWQ82I 134148676 IC50 = 220 nM T46781 CN7FJ9 134149620 IC50 = 48 nM T46781 CFZ7J9 134152243 IC50 = 28 nM T46781 CIP61L 134153498 EC50 = 7.1 nM T46781 CXT13L 134154154 IC50 = 32 nM T46781 CFN7Q8 134156381 IC50 = 15 nM T46781 CQ07HK 134157266 IC50 = 30 nM T46781 COK96J 134827795 IC50 = 23700 nM T46781 CIZ39M 134827836 IC50 > 100000 nM T46781 CJ04NP 134827837 IC50 > 100000 nM T46781 CGBZ13 134843302 IC50 = 900 nM T46781 C54FXD 134957362 IC50 > 10000 nM T46781 CS4OW8 135400873 IC50 = 815 nM T46781 CJ65LQ 135423783 IC50 > 100000 nM T46781 C2WL8M 135423784 IC50 > 100000 nM T46781 CNKD13 135423790 IC50 = 7000 nM T46781 C48NWF 135423791 IC50 = 8000 nM T46781 CEVL69 135423792 IC50 = 4600 nM T46781 C6HGC3 135423793 IC50 = 10000 nM T46781 C1W6EI 135423851 IC50 > 100000 nM T46781 CYH51Q 135423852 IC50 > 100000 nM T46781 CYG2V6 135428039 IC50 = 2.6 nM T46781 CK9D4A 135428921 IC50 = 59 nM T46781 CUFC14 135502940 IC50 = 130 nM T46781 C9ZBY3 135525654 IC50 = 150 nM T46781 CTB7R2 135564980 IC50 = 5 nM T46781 C6QA2T 135566358 IC50 = 75 nM T46781 CJN0Z7 135566360 IC50 = 54 nM T46781 CZY5G2 135566361 IC50 = 180 nM T46781 C7PJ6X 135566704 IC50 = 275 nM T46781 CF0CM3 135909510 IC50 = 510 nM T46781 CVH9A7 135909511 IC50 = 15 nM T46781 CWIE69 135909512 IC50 = 10 nM T46781 CGSC82 135909513 IC50 = 5.2 nM T46781 CQ1RH0 135909514 IC50 = 24 nM T46781 CX02VW 135909515 IC50 = 10 nM T46781 C8VU0O 135929094 IC50 = 220 nM T46781 CEP9Y5 135929097 IC50 = 510 nM T46781 C9N3GW 135929098 IC50 = 880 nM T46781 CVG4I5 135929100 IC50 = 2 nM T46781 C0V2HQ 135929101 IC50 = 86 nM T46781 C01HMT 135932346 IC50 = 24 nM T46781 CIPA79 135937899 IC50 = 4200 nM T46781 C2PAV1 135971426 IC50 = 640 nM T46781 C4RL7Q 135985508 IC50 = 210 nM T46781 CHA4N2 136013680 IC50 > 10 nM T46781 C3I2CY 136065819 IC50 = 1580 nM T46781 CAW0E4 136065882 IC50 = 227 nM T46781 C21PTY 136104462 IC50 > 100000 nM T46781 C7XO8B 136104463 IC50 > 100000 nM T46781 C7UH8T 136104464 IC50 > 100000 nM T46781 C7R2PD 136104467 IC50 > 100000 nM T46781 CLEN23 136104468 IC50 > 100000 nM T46781 CWLJ05 136104469 IC50 > 100000 nM T46781 CRI97Z 136126922 IC50 = 91.8 nM T46781 CZUP29 136126923 IC50 = 143.9 nM T46781 CFZ50A 136126924 IC50 = 412.3 nM T46781 C2THI7 136126927 IC50 = 191 nM T46781 CG90AI 136126928 IC50 = 138.6 nM T46781 CKU26Y 136126929 IC50 = 231.3 nM T46781 CQ6PT9 136126930 IC50 = 424.1 nM T46781 C4R0ET 136126935 IC50 = 1201 nM T46781 CQI7M9 136126936 IC50 = 98.8 nM T46781 CWJY91 136126938 IC50 = 2.2 nM T46781 CW4JI1 136126939 IC50 = 2.3 nM T46781 CZ7EX0 136183413 IC50 = 270 nM T46781 C6HW4E 136206295 IC50 = 11100 nM T46781 CU9P3M 136206296 IC50 = 7000 nM T46781 C1YUD0 136219394 IC50 > 10 nM T46781 C8UH0A 136226786 IC50 > 10000 nM T46781 CU62DL 136234658 IC50 = 392.3 nM T46781 CIU8W3 136254389 IC50 > 10 nM T46781 CFQO70 136375226 IC50 = 35 nM T46781 C3MK9W 136807986 IC50 > 10000 nM T46781 CB6G3P 136966265 IC50 > 10000 nM T46781 CH3M4B 137083628 IC50 > 30000 nM T46781 CJA07O 137083629 IC50 > 30000 nM T46781 C9F8PX 137083630 IC50 > 30000 nM T46781 CXC69T 137321158 IC50 = 210 nM T46781 CAI3O8 137633471 IC50 = 250 nM T46781 C3WUN4 137633742 IC50 > 100000 nM T46781 C1X2EL 137634130 IC50 > 100000 nM T46781 CI1E8V 137634241 IC50 > 10000 nM T46781 CPF75D 137636602 IC50 > 100000 nM T46781 C8C6HP 137637035 IC50 = 1200 nM T46781 CA8GF2 137637401 IC50 = 229 nM T46781 C2L3HG 137637474 IC50 = 9000 nM T46781 CO6I5H 137637664 IC50 > 100000 nM T46781 CSGZ41 137638900 IC50 > 100000 nM T46781 C21QTU 137639046 IC50 = 2300 nM T46781 C5LYA1 137639191 IC50 = 6200 nM T46781 CE96AL 137639657 IC50 = 6200 nM T46781 C6U5BY 137640035 IC50 = 460 nM T46781 CZS13Q 137640111 IC50 = 959 nM T46781 CN92SG 137640413 IC50 > 100000 nM T46781 CHB5Z8 137643106 IC50 = 270 nM T46781 C2VTY1 137643199 IC50 = 3000 nM T46781 CV54HX 137643853 IC50 = 360 nM T46781 CESF45 137644276 IC50 = 853 nM T46781 CD29JK 137644944 IC50 > 100000 nM T46781 C9GIO5 137645634 IC50 = 1000 nM T46781 CP85WU 137646574 IC50 = 51000 nM T46781 CQOL75 137646726 IC50 = 270 nM T46781 CZO42N 137648629 IC50 > 100000 nM T46781 C0VSY4 137648758 IC50 = 120 nM T46781 CF7Y1Z 137649033 IC50 > 100000 nM T46781 C0C9SG 137649545 IC50 > 100000 nM T46781 C3LAD6 137652990 IC50 > 100000 nM T46781 CZ2QG8 137654305 IC50 > 100000 nM T46781 CE3AM1 137654624 IC50 = 90 nM T46781 CRH18Z 137656846 IC50 = 1345 nM T46781 CA9K8C 137657902 IC50 = 110 nM T46781 CI2R1O 137658474 IC50 = 1400 nM T46781 CO41NV 137658479 IC50 > 100000 nM T46781 CLTJ12 137658608 IC50 > 100000 nM T46781 C7G2KR 137659019 IC50 = 320 nM T46781 CWXL97 137659452 IC50 = 700 nM T46781 C98HDI 137660135 IC50 = 3100 nM T46781 CLN6C1 137662100 IC50 = 700 nM T46781 CM3UF7 137700779 IC50 > 10000 nM T46781 CQR52I 141143841 IC50 = 13 nM T46781 C7GR6C 141483894 IC50 = 11500 nM T46781 C0NP3Z 141483896 IC50 > 100000 nM T46781 C1RD0T 145949228 IC50 = 102.3 nM T46781 C4RL0N 145949878 IC50 = 121.5 nM T46781 CH9YZ4 145949906 IC50 > 1000 nM T46781 CTH9R6 145950406 IC50 = 89.2 nM T46781 C4TB3R 145950483 IC50 = 526.1 nM T46781 C95UCZ 145950577 IC50 = 86.1 nM T46781 C2NA5J 145950876 IC50 = 34.6 nM T46781 C07HDJ 145951056 IC50 = 352.5 nM T46781 C8FPE7 145951250 IC50 = 335.9 nM T46781 C7ED9I 145952622 IC50 = 657.1 nM T46781 CHBF06 145952797 IC50 = 74.9 nM T46781 CN2VT9 145953211 IC50 = 25.7 nM T46781 CLA54T 145954009 IC50 = 945.9 nM T46781 CZ7I2Y 145954624 IC50 = 102 nM T46781 C9HUW7 145955353 IC50 = 66.2 nM T46781 C9VXM4 145955906 IC50 = 73.3 nM T46781 C3IH0W 145956084 IC50 = 835.2 nM T46781 C8WIA4 145957055 IC50 = 700.3 nM T46781 CE90PN 145957225 IC50 = 442 nM T46781 C1JDL3 145957276 IC50 = 121.6 nM T46781 CUI3W1 145957403 IC50 = 101 nM T46781 CLDG46 145957722 IC50 > 1000 nM T46781 CC10SH 145958079 IC50 = 188 nM T46781 C89XYV 145958579 IC50 = 145 nM T46781 C2W9IL 145959003 IC50 = 75.1 nM T46781 CV08DO 145959172 IC50 = 140.4 nM T46781 C70IJE 145959540 IC50 = 83.6 nM T46781 C1U8PV 145959596 IC50 > 1000 nM T46781 C7M6XN 145960087 IC50 = 452 nM T46781 C8VPI4 145960125 IC50 = 60.2 nM T46781 CT30CG 145960449 IC50 > 10000 nM T46781 CE9D6T 145960511 IC50 > 10000 nM T46781 C4M6SJ 145961986 IC50 > 10000 nM T46781 CQE9M5 145966810 IC50 = 170 nM T46781 CK4IV6 145967934 IC50 = 105 nM T46781 CD58LC 145967944 IC50 = 132 nM T46781 CDNC31 145967951 IC50 < 13 nM T46781 C75HDR 145968148 IC50 < 13 nM T46781 C0DEU9 145968159 IC50 < 13 nM T46781 CY7FL8 145968605 EC50 < 16 nM T46781 CRAL38 145968638 IC50 < 13 nM T46781 CRD0G4 145969024 IC50 < 13 nM T46781 CWJ12M 145969155 IC50 = 100 nM T46781 CCH2R0 145969234 IC50 = 80 nM T46781 CL9F4K 145969442 IC50 < 13 nM T46781 C23VZS 145969582 IC50 = 134 nM T46781 CX70KC 145969955 IC50 < 13 nM T46781 CY43DF 145970132 IC50 < 13 nM T46781 CIOX52 145970381 IC50 < 13 nM T46781 CQY4I3 145970473 IC50 < 13 nM T46781 CPO34H 145970612 IC50 < 13 nM T46781 C8WX1F 145970663 IC50 < 13 nM T46781 CA03CS 145970720 IC50 < 13 nM T46781 CJ59ZQ 145970874 IC50 = 265 nM T46781 CT73QK 145971147 IC50 < 13 nM T46781 CI9B2A 145971241 IC50 = 78.9 nM T46781 CUW6I0 145972008 IC50 = 443 nM T46781 C54FIC 145979195 IC50 = 17 nM T46781 C9DE2V 145979557 IC50 = 2320.6 nM T46781 CYH41T 145979752 IC50 = 4594 nM T46781 CLU75C 145979974 IC50 = 41 nM T46781 CX63VM 145980115 IC50 = 278.1 nM T46781 CUA34Y 145980364 IC50 = 1271 nM T46781 C05GKB 145980665 IC50 > 100000 nM T46781 CNS6I5 145980673 IC50 = 854.4 nM T46781 CR0JD7 145981097 IC50 = 611 nM T46781 CU25SM 145981644 IC50 = 321.6 nM T46781 C7AE4L 145981787 IC50 = 2522 nM T46781 C5YCJ0 145982003 IC50 = 37.6 nM T46781 CDB3X6 145982088 IC50 = 773 nM T46781 CQ8A6B 145982177 IC50 = 50.3 nM T46781 CVES49 145982552 IC50 > 10000 nM T46781 CJ8Y9M 145982688 IC50 = 11 nM T46781 CIDU48 145982789 IC50 > 10000 nM T46781 CPO43Z 145982872 IC50 > 10000 nM T46781 CORV50 145982985 IC50 > 10000 nM T46781 C6YBK0 145983031 IC50 > 10000 nM T46781 CD3WR9 145983454 IC50 > 10000 nM T46781 CQXC48 145983553 IC50 > 10000 nM T46781 CJ4N1S 145983820 IC50 > 10000 nM T46781 C8GVD0 145984001 IC50 > 10000 nM T46781 CG0B6W 145984157 IC50 > 60000 nM T46781 CTJW32 145984202 IC50 > 10000 nM T46781 C8C5XL 145984893 IC50 = 31 nM T46781 C48YNJ 145985058 IC50 > 10000 nM T46781 C67EVF 145985214 IC50 > 10000 nM T46781 CKQ69G 145985465 IC50 > 10000 nM T46781 C9WDL3 145986316 IC50 = 54.1 nM T46781 CE05UV 145986353 IC50 < 13 nM T46781 C64JZF 145986550 IC50 = 6282 nM T46781 C8NDE5 145987193 IC50 = 547 nM T46781 C76OKW 145987254 IC50 = 1147 nM T46781 C1BR4S 145987787 IC50 = 893 nM T46781 C7LV2F 145987970 IC50 = 86 nM T46781 CWYN61 145988204 IC50 = 35 nM T46781 C8XD0B 145988239 IC50 = 1003.6 nM T46781 C6S8BD 145988336 IC50 = 417 nM T46781 C61BLV 145988464 IC50 > 100000 nM T46781 CSWQ20 145988550 IC50 = 270 nM T46781 C1NS8U 145989128 IC50 = 23 nM T46781 C5EZ1P 145989138 IC50 = 2681.5 nM T46781 C0GNE7 145989369 IC50 = 352 nM T46781 CT9D0X 145989541 IC50 = 1620 nM T46781 CI3B9F 145989892 IC50 = 307.4 nM T46781 CFM97W 145990241 IC50 = 610.5 nM T46781 C5NB4O 145990292 IC50 = 29 nM T46781 C9T1UF 145990998 IC50 = 38 nM T46781 CQU8G2 145991240 IC50 = 48 nM T46781 CKE21U 145991373 IC50 = 127 nM T46781 CAK5V0 145992869 IC50 = 1184.7 nM T46781 CG27SA 145993108 IC50 = 46 nM T46781 C0AHF1 145993112 IC50 = 14360 nM T46781 CE7M4S 145993303 IC50 > 100000 nM T46781 C0YA9U 145993477 IC50 = 894 nM T46781 CS3DY6 145993716 IC50 = 99.8 nM T46781 C2MD1Q 155513187 IC50 = 1239 nM T46781 CZEO50 155513953 IC50 = 63.1 nM T46781 C2NB1R 155514901 IC50 = 3.5 nM T46781 CJD0Z2 155515276 IC50 = 3.07 nM T46781 C0PG3L 155516058 IC50 = 2.8 nM T46781 C7VB6R 155516420 IC50 = 0.34 nM T46781 CM45EF 155519065 IC50 = 3.5 nM T46781 CM0IC7 155521232 IC50 = 5011.87 nM T46781 CEA2C1 155521505 IC50 = 1.11 nM T46781 C2EHI7 155524928 IC50 = 1584.89 nM T46781 C1STO9 155525257 IC50 = 0.29 nM T46781 C52FHM 155525581 IC50 = 19.5 nM T46781 CDZ59A 155527907 IC50 = 27 nM T46781 C0DZ9X 155527985 IC50 = 79.43 nM T46781 CFR56S 155533031 IC50 = 316.23 nM T46781 C90SIO 155535101 IC50 = 2.67 nM T46781 C9JD7A 155535968 IC50 = 100 nM T46781 C2CG1A 155537016 IC50 > 10000 nM T46781 C68GMW 155538446 IC50 = 7800 nM T46781 CT9IM4 155539207 IC50 = 8530 nM T46781 CM4I2F 155540641 IC50 = 0.67 nM T46781 CTG40B 155541947 IC50 = 3.29 nM T46781 C9T1YR 155543136 IC50 = 11.3 nM T46781 CC5P1X 155543762 IC50 = 17.3 nM T46781 CF1AJ2 155544000 IC50 = 199.53 nM T46781 C27GLF 155545018 IC50 = 49.1 nM T46781 CY6Q8S 155554337 IC50 = 31000 nM T46781 CIY5U0 155556737 IC50 = 100 nM T46781 C9XK2G 155559311 IC50 = 2.55 nM T46781 CO2I4P 155559898 IC50 = 800 nM T46781 COSE65 155561444 IC50 = 1995.26 nM T46781 C13GYL 127031746 IC50 < 5000 nM T46781 D00HVA 11624601 Ki > 6700 nM T46781 D00JMT 210332 IC50 = 75 nM T46781 D00UTU 136104465 IC50 = 20000 nM T46781 D01YWE 25207521 IC50 = 1400 nM T46781 D03BJF 44465558 IC50 = 700 nM T46781 D03DZO 11715767 IC50 > 10000 nM T46781 D03YVL 5472558 IC50 = 15600 nM T46781 D04MYT 46885627 IC50 = 13398 nM T46781 D04NGS 5330790 IC50 = 4 nM T46781 D04WFN 10202471 IC50 = 35 nM T46781 D04YQF 763936 IC50 = 6500 nM T46781 D06AGN 136043837 IC50 = 2100 nM T46781 D06LJL 9916282 IC50 = 7 nM T46781 D06QWO 14824655 IC50 > 10 ug.mL-1 T46781 D07ADX 54764565 IC50 = 123 nM T46781 D08HFG 24809764 IC50 > 10000 nM T46781 D09HVH 135566652 IC50 > 10 nM T46781 D09KEB 11493841 IC50 = 3981.07 nM T46781 D0A1CM 5281855 IC50 = 2500 nM T46781 D0A7FQ 11644425 IC50 = 2500 nM T46781 D0AY0F 70698427 IC50 > 10000 nM T46781 D0CE3R 5312137 IC50 = 19 nM T46781 D0EU1R 46215815 IC50 = 3162.28 nM T46781 D0G3SZ 6918469 IC50 = 1.1 ug.mL-1 T46781 D0I1IK 136104466 IC50 = 8000 nM T46781 D0IZ8M 56675928 IC50 = 2252 nM T46781 D0ME9B 46868971 IC50 <= 13 nM T46781 D0N4LR 53469448 IC50 = 407 nM T46781 D0Q3NG 11715520 Ki > 6700 nM T46781 D0Q7TO 6419766 IC50 = 858 nM T46781 D0QC0W 9914412 IC50 = 51 nM T46781 D0S3RP 135458003 IC50 > 30000 nM T46781 D0S7IE 11658882 Ki > 6700 nM T46781 D0T4SJ 10356352 IC50 = 2140 nM T46781 D0U8VY 6610278 IC50 = 1250 nM T46781 D0V6LP 136043836 IC50 = 3000 nM T46781 D0Y0ES 3707 IC50 = 2300 nM T83875 D01ZSO 4235 Ki = 5 nM T83875 D03GET 4055 Ki = 26000 nM T83875 D04AIT 5280445 IC50 = 4900 nM T83875 D06OMW 3052776 IC50 = 587 nM T83875 D07UYO 441401 IC50 = 8.1 ug.mL-1 T83875 D08KBK 11234049 Ki < 2000 nM T83875 D08SKH 4114 IC50 = 85110 nM T83875 D09QDP 4380 IC50 = 0.0049 nM T83875 D0B3HD 2519 IC50 > 50000 nM T83875 D0E7PQ 5311 IC50 > 100000 nM T83875 D0H0HJ 19493 IC50 = 1020 nM T83875 D0J2MJ 26758 IC50 = 1700 nM T83875 D0K8KX 5280343 IC50 = 2440 nM T83875 D0NS6H 3152 IC50 = 850000 nM T83875 D0P9AC 3675 Ki = 163 nM T83875 D0R0UJ 4688 IC50 = 1310 nM T83875 D0S2UG 26757 IC50 = 67.25 nM T83875 D0T1LK 4908 IC50 = 75700 nM T83875 D0T3LF 5826 Ki = 14400 nM T83875 D0TV6I 131682 IC50 = 25900 nM T83875 D00VUI 6199 IC50 > 20000 nM T83875 D05PCM 78323835 IC50 = 6000 nM T83875 D07SDQ 969516 Ki = 710 nM T83875 D0C3UC 208907 IC50 = 85000 nM T83875 D0DI6L 11476460 IC50 = 1.8 ug.mL-1 T83875 D0H7PW 638024 IC50 = 58980 nM T83875 D0I2GS 25184541 IC50 = 41.9 ug.mL-1 T83875 D0I4ZN 66571643 IC50 > 100000 nM T83875 D0L4FS 5280961 IC50 = 3900 nM T83875 D0LI1C 44469321 IC50 > 10000 nM T83875 D0QR5G 2355 IC50 = 13800 nM T83875 D0U3EP 445154 IC50 = 15700 nM T83875 D0W7LO 9947954 IC50 = 287.3 nM T83875 D00OWF 5280953 Ki = 5 nM T83875 D02EME 137653313 IC50 = 4600 nM T83875 D02FRR 77844720 IC50 > 10000 nM T83875 D04AXC 46829776 IC50 = 8600 nM T83875 D06BFA 77844660 IC50 > 10000 nM T83875 D06QRW 71307 IC50 > 80000 nM T83875 D08YYW 77844717 IC50 > 10000 nM T83875 D0AF7J 77844718 IC50 = 0.6607 nM T83875 D0K2LB 77844666 IC50 < 10000 nM T83875 D0NB7Z 46829772 IC50 = 4900 nM T83875 D0R6RT 137652717 IC50 = 3400 nM T83875 D0RN2X 442126 IC50 = 1760 nM T83875 D0U9TR 53262706 IC50 > 100000 nM T83875 D0UL2R 77844722 Ki = 0.48 nM T83875 D01LAC 6437850 Ki = 1100 nM T83875 D0E8UJ 126111 Ki = 10 nM T83875 D0IZ1D 44571 IC50 = 180 nM T83875 C2ZB4C 5530 IC50 = 4720 nM T83875 CK4N7S 6293 IC50 = 30100 nM T83875 CV6BH8 6809 IC50 = 165000 nM T83875 CI8X6J 6885 IC50 = 44900 nM T83875 C5QAH4 7020 IC50 = 840 nM T83875 CJD54S 7578 Ki = 7720 nM T83875 C1G4XA 8764 Ki = 24100 nM T83875 CP0O8I 9513 Ki = 121400 nM T83875 CSCE03 9688 IC50 = 5030 nM T83875 CUV23A 10286 IC50 = 39900 nM T83875 C5SRE2 10658 Ki = 460 nM T83875 C8H4SX 10724 IC50 = 14800 nM T83875 C5NKT4 15362 Ki = 27000 nM T83875 C9FEQ0 16717 Ki = 18100 nM T83875 C0PFU5 21107 IC50 > 100000 nM T83875 C3YEH9 22652 Ki = 4000 nM T83875 C6IN5F 22860 Ki = 50300 nM T83875 C2N0TD 26070 IC50 = 3400 nM T83875 C3IEL1 26861 IC50 > 100000 nM T83875 C3VL1J 27694 Ki = 27000 nM T83875 CBSV68 37764 Ki = 1300000 nM T83875 CA98UO 40010 Ki = 77000 nM T83875 C3RM6D 46697 Ki = 34000 nM T83875 C64WMG 52356 IC50 = 15200 nM T83875 C09AHX 68081 IC50 > 20000 nM T83875 CBP13T 69512 IC50 = 22100 nM T83875 CT8ZH3 71034 IC50 = 5300 nM T83875 C6UKD8 74342 IC50 = 45600 nM T83875 CT7HM1 74708 IC50 = 3800 nM T83875 CQ94EN 77309 IC50 = 180 nM T83875 CZY6R3 78027 Ki = 5700 nM T83875 CA60QP 81046 IC50 = 900 nM T83875 CMQ6U7 81528 Ki = 2300 nM T83875 CB04TP 83054 Ki = 34500 nM T83875 CSU27D 83242 Ki = 31000 nM T83875 CQ1RK5 87112 IC50 = 28900 nM T83875 C3P1QX 88562 Ki = 3000 nM T83875 C5HO0S 92892 Ki = 123000 nM T83875 CK1H3L 97662 IC50 > 20000 nM T83875 C4VE6D 99562 IC50 > 10000 nM T83875 C0N9VI 100742 IC50 = 65250 nM T83875 CIF4J3 114679 IC50 = 6200 nM T83875 C01QZU 127234 IC50 > 100000 nM T83875 C6L0WU 133354 IC50 = 9700 nM T83875 CZ15VX 134885 IC50 > 200000 nM T83875 CSU36M 136620 IC50 = 38930 nM T83875 C8W9IH 138472 Ki = 93500 nM T83875 CZ45BJ 147354 IC50 > 100000 nM T83875 CUZN14 156448 Ki = 260000 nM T83875 C1ND9W 161665 IC50 > 20000 nM T83875 CFJ52D 164751 Ki = 186000 nM T83875 C2QHX7 177014 IC50 > 20000 nM T83875 C1CEJ8 182118 IC50 > 100000 nM T83875 CF43TE 199605 IC50 = 68730 nM T83875 CXE58T 217219 IC50 > 100000 nM T83875 CW8R2J 223515 Ki = 24270 nM T83875 C69FVR 223547 Ki = 9570 nM T83875 CACH74 223561 Ki = 26320 nM T83875 CNL5A0 223570 Ki = 5570 nM T83875 C6PDH2 252679 IC50 = 67.61 nM T83875 C3A9FD 255751 IC50 = 6480 nM T83875 CDB2W6 267093 Ki = 6450 nM T83875 CBM9H4 275641 IC50 = 1390 nM T83875 COGF79 300241 IC50 = 30000 nM T83875 C3E1TC 304813 IC50 = 51630 nM T83875 C4PUL2 343657 IC50 = 45200 nM T83875 C5RMJ2 347809 IC50 > 100000 nM T83875 CE8CT9 352026 IC50 = 56400 nM T83875 C69DUA 352028 IC50 = 8220 nM T83875 CS2F1T 371801 IC50 = 3580 nM T83875 CJ48SW 420804 Ki = 36000 nM T83875 C7HME8 439246 IC50 = 955000 nM T83875 C8N6PO 442186 Ki = 102000 nM T83875 CYB16H 442356 Ki = 160000 nM T83875 CB32AN 473589 IC50 = 6260 nM T83875 CP7Y4O 476960 Ki = 950 nM T83875 CIS41L 479656 IC50 = 51000 nM T83875 CMT3P0 480764 IC50 = 38800 nM T83875 C14AWI 499408 Ki = 37000 nM T83875 C7N6MD 580653 IC50 = 93600 nM T83875 CK1J3F 602830 Ki = 1430 nM T83875 C8M1SX 605698 Ki = 13000 nM T83875 C2KHP1 605727 Ki = 80000 nM T83875 CV36NW 607796 IC50 = 5370 nM T83875 CZ4OC0 611428 IC50 = 1300 nM T83875 C8HRD3 613011 Ki = 41000 nM T83875 COVU71 613852 Ki = 700000 nM T83875 CO0H7W 621883 Ki = 17000 nM T83875 C4VIH5 636991 IC50 = 27320 nM T83875 C2IRO1 638256 IC50 > 20000 nM T83875 C0C7MF 641818 IC50 > 100000 nM T83875 C4KYW6 649393 IC50 = 42320 nM T83875 CD8KC2 673374 IC50 > 100000 nM T83875 CP91NX 677915 IC50 = 19800 nM T83875 CZ7XE1 680623 IC50 > 100000 nM T83875 C5QIK2 682145 IC50 > 100000 nM T83875 CPIT91 682187 IC50 = 35510 nM T83875 CDE9V2 689424 IC50 = 48100 nM T83875 C5O0TJ 690158 IC50 = 82800 nM T83875 CM51LR 692546 IC50 > 100000 nM T83875 CUHY04 692606 IC50 > 100000 nM T83875 C46VZA 692702 IC50 > 100000 nM T83875 C61FYO 693313 IC50 = 64800 nM T83875 CQV73I 694612 IC50 = 13060 nM T83875 CT9R3F 694735 IC50 > 100000 nM T83875 CC40ZA 711807 IC50 = 4800 nM T83875 CU4IZ0 724176 IC50 = 15140 nM T83875 CVJ15O 724191 IC50 = 12320 nM T83875 CQ59DC 724193 IC50 = 15950 nM T83875 C3YOJ2 724194 IC50 = 20630 nM T83875 C2NVT7 724195 IC50 = 18770 nM T83875 CIS57F 724196 IC50 = 17560 nM T83875 C9NYF1 728520 IC50 = 2620 nM T83875 C6SQ9Y 735483 IC50 = 42500 nM T83875 C8J0PG 737170 IC50 > 100000 nM T83875 C54GJN 747648 IC50 = 346.74 nM T83875 CL9GS4 764149 IC50 = 2550 nM T83875 CTRO75 781371 IC50 = 61460 nM T83875 C2U0LO 794222 IC50 > 100000 nM T83875 C27LMJ 797192 IC50 = 9450 nM T83875 CAKL20 807313 IC50 > 100000 nM T83875 CDU38G 834420 Ki = 1540 nM T83875 CK2Z1F 852572 IC50 = 42400 nM T83875 CGCD65 871734 IC50 > 100000 nM T83875 CF89IZ 872422 IC50 = 9790 nM T83875 CYVA98 874919 IC50 = 16700 nM T83875 C72NHE 877852 IC50 = 550 nM T83875 C3XY5A 882744 IC50 = 1120 nM T83875 CSX7H6 882845 IC50 = 6770 nM T83875 C6GM0Z 886539 IC50 = 50 nM T83875 COUL71 891711 IC50 = 64200 nM T83875 CQ4I9A 894713 IC50 > 100000 nM T83875 CIN30B 894965 IC50 = 48700 nM T83875 C02WCM 895200 IC50 = 39700 nM T83875 CC8IJ5 895343 IC50 = 88300 nM T83875 C0MS5E 927669 IC50 > 50000 nM T83875 CZFU46 958268 IC50 = 3520 nM T83875 CUMA52 965710 IC50 = 17782.79 nM T83875 CIT3L2 1016023 IC50 = 7910 nM T83875 C4YAE7 1037029 IC50 = 37900 nM T83875 C5S2LQ 1178193 IC50 = 17700 nM T83875 CKFO95 1201119 IC50 = 67310 nM T83875 C47DQB 1211950 IC50 > 100000 nM T83875 C82HEY 1241457 IC50 = 5430 nM T83875 C7EGD5 1249836 IC50 = 1040 nM T83875 CA84HD 1251882 IC50 = 2770 nM T83875 CDVS56 1268920 IC50 = 28550 nM T83875 C9G1NF 1269411 IC50 = 39890 nM T83875 CF7GZ3 1272788 Ki = 6670 nM T83875 CA9U8F 1332620 IC50 > 10000 nM T83875 C0IHA6 1345219 IC50 = 35260 nM T83875 CA0B1Y 1381460 IC50 = 21800 nM T83875 CBW19M 1383560 IC50 = 35260 nM T83875 CZ47DC 1397819 IC50 = 12970 nM T83875 CED0S4 1416314 IC50 = 70500 nM T83875 CCX9O4 1489242 Ki = 719448978 nM T83875 C4AR3X 1494342 IC50 = 27900 nM T83875 CM80QJ 1509337 IC50 = 4700 nM T83875 CENL04 1523065 IC50 = 979 nM T83875 C9TR4H 1523287 IC50 = 49070 nM T83875 CL9UE7 1641788 IC50 = 43460 nM T83875 CM02NF 1712168 IC50 = 398800 nM T83875 COB92M 1730869 IC50 = 685000 nM T83875 CBR10Z 1773356 IC50 = 39360 nM T83875 CQR67C 1909002 Ki = 8140 nM T83875 CW4G6A 1929998 IC50 = 10580 nM T83875 CQSP80 2237121 IC50 > 100000 nM T83875 CM5XN1 2329351 IC50 = 29850 nM T83875 CF81QZ 2629406 IC50 = 240 nM T83875 CEQ4V8 2723716 IC50 = 10600 nM T83875 CO3JT6 2728600 IC50 > 100000 nM T83875 C61MIZ 2737276 IC50 > 100000 nM T83875 C9AH7R 2774040 IC50 = 161000 nM T83875 C3QHE9 2785758 IC50 = 183000 nM T83875 CCH4L0 2798381 IC50 = 40360 nM T83875 CNP4S1 2806094 IC50 > 100000 nM T83875 C2EL5W 2826990 Ki = 6000 nM T83875 CANM16 2827498 IC50 = 5360 nM T83875 C8RBP0 2888531 IC50 = 43020 nM T83875 C0E7TW 3035046 IC50 > 200000 nM T83875 C2XP0H 3052775 IC50 = 710 nM T83875 C4DCJ7 3082143 Ki = 87000 nM T83875 CKD72T 3083848 IC50 = 1780 nM T83875 CR7AK6 3132916 IC50 = 67300 nM T83875 CC48UQ 3162481 IC50 > 10000 nM T83875 C2GE9F 3162506 IC50 > 10000 nM T83875 CLFE62 3333374 IC50 = 273000 nM T83875 C6IPM8 3391493 IC50 = 100 nM T83875 CX7T5S 3517936 IC50 > 100000 nM T83875 CEM29H 3547496 Ki = 14996848.36 nM T83875 C90THR 3553261 IC50 > 100000 nM T83875 C5DV0S 3596769 IC50 = 28200 nM T83875 CCW40J 3670544 IC50 = 54954.09 nM T83875 CX0AD8 3778700 IC50 = 51600 nM T83875 C9M3YA 3811175 IC50 = 43000 nM T83875 CR9Y4X 3928946 IC50 = 41400 nM T83875 C18AYX 4313470 Ki = 5100 nM T83875 CMEC57 4539762 IC50 > 500000 nM T83875 C70WJL 4679494 IC50 = 43800 nM T83875 CFQ3J7 4779843 IC50 = 550 nM T83875 CT6GY3 5169444 IC50 = 14200 nM T83875 C84CKE 5200299 IC50 = 89600 nM T83875 CWE84I 5281233 IC50 = 170000 nM T83875 CL1MR9 5281254 Ki = 100 nM T83875 C3OVR2 5281623 IC50 = 660 nM T83875 CAEF10 5281626 IC50 = 13000 nM T83875 CE6K3P 5281635 IC50 = 8000 nM T83875 C3B2WJ 5281651 IC50 = 40 nM T83875 CH01XT 5281656 IC50 = 25000 nM T83875 CBD68R 5281658 IC50 = 24000 nM T83875 CTA0N2 5281661 IC50 = 8500 nM T83875 CLZ3Q1 5281663 IC50 = 3800 nM T83875 CE5SI3 5281725 IC50 = 11250 nM T83875 CBUL97 5281728 IC50 = 19600 nM T83875 C5LGJ1 5282362 IC50 > 100000 nM T83875 CQ7TV2 5314262 IC50 = 13200 nM T83875 CPRI38 5320318 Ki = 260 nM T83875 CC7RD0 5320946 IC50 = 51 nM T83875 C2IZ9D 5322196 IC50 = 48200 nM T83875 CEG8R3 5322280 IC50 = 60110 nM T83875 CNA80W 5337609 Ki = 240 nM T83875 CXCI17 5345068 IC50 = 1650 nM T83875 C9D5NA 5346030 IC50 > 100000 nM T83875 CXKD41 5348419 IC50 > 100000 nM T83875 CPW0G3 5354554 IC50 > 100000 nM T83875 CW6IE0 5356384 IC50 > 100000 nM T83875 C8ZJ2Q 5357659 Ki = 100 nM T83875 C54BYP 5360741 IC50 = 1710 nM T83875 C8GT7Y 5366975 IC50 = 4300 nM T83875 C7EZA1 5368282 IC50 = 3650 nM T83875 C7FCX1 5370710 IC50 = 297000 nM T83875 C4S1UA 5375423 Ki = 8010 nM T83875 C1EKB8 5376013 IC50 = 1100 nM T83875 C70YLN 5376036 IC50 = 310 nM T83875 CO6JI8 5377044 IC50 = 3700 nM T83875 CM3T9J 5377817 IC50 > 100000 nM T83875 C7AE9W 5378284 IC50 = 19000 nM T83875 C4T1CZ 5388521 IC50 = 1520 nM T83875 C1HKU6 5464639 IC50 = 65000 nM T83875 C8QP4J 5467625 IC50 = 709 nM T83875 CCUM24 5467627 IC50 = 268 nM T83875 CXM6S3 5479773 IC50 = 29000 nM T83875 CL4CM3 5480299 IC50 = 730 nM T83875 C5O9YH 5480342 IC50 = 2700 nM T83875 CH1G9B 5480343 IC50 = 32000 nM T83875 C9YB8H 5480344 IC50 = 51000 nM T83875 CWO9S6 5491377 IC50 = 110 nM T83875 CME0C2 5709307 IC50 = 41800 nM T83875 C1QUA7 5711036 IC50 > 10000 nM T83875 CRQ3P9 5711038 IC50 > 10000 nM T83875 C26HRP 5717651 IC50 = 18600 nM T83875 C8A3JH 5717653 IC50 = 24000 nM T83875 C6SR2J 5718033 IC50 = 85700 nM T83875 C7IZJ1 5723719 IC50 > 100000 nM T83875 CKN25F 5727970 IC50 = 1550 nM T83875 CZ79RX 5728224 Ki = 560 nM T83875 CM7V8F 5729327 Ki = 600 nM T83875 CVM37E 5731408 IC50 = 19200 nM T83875 CCM41G 5780273 Ki = 240 nM T83875 CW0M9V 5784792 IC50 > 100000 nM T83875 CU1I8E 5815007 IC50 = 4060 nM T83875 C2F4QH 5820198 IC50 = 3490 nM T83875 C7TOI9 5863209 IC50 > 100000 nM T83875 CE59LJ 5908055 Ki = 140 nM T83875 CK0M4A 5910585 IC50 = 26915.35 nM T83875 CJS0P7 5945471 IC50 > 100000 nM T83875 CFN9G8 5989034 IC50 > 100000 nM T83875 C5V4SY 6093310 Ki = 70000 nM T83875 C73HMS 6106285 Ki = 160 nM T83875 CL9Z1S 6110591 Ki = 130 nM T83875 C31OYT 6163838 Ki = 490 nM T83875 CYX45A 6213016 IC50 > 100000 nM T83875 CT8N5B 6370756 IC50 = 520 nM T83875 CP0XL9 6419979 Ki = 284000 nM T83875 C40RHI 6421573 IC50 = 157100 nM T83875 CFWP52 6433444 IC50 > 10000 nM T83875 C1N0KP 6436743 Ki = 970 nM T83875 CEKT60 6438383 Ki = 231000 nM T83875 C1VU0Y 6461059 IC50 > 100000 nM T83875 CRDF19 6474563 IC50 > 10000 nM T83875 CGHV31 6864775 IC50 = 4990 nM T83875 CNL1X8 6873295 IC50 > 10000 nM T83875 CUJA07 6896171 IC50 > 10000 nM T83875 CO6SY2 7061238 Ki = 6000 nM T83875 C30EFO 7157331 Ki = 31000 nM T83875 C5L8EP 7214067 IC50 > 10000 nM T83875 CL95KF 7245716 IC50 = 59610 nM T83875 CM91LR 7559290 IC50 > 10000 nM T83875 CI4NS5 7695078 IC50 = 5980 nM T83875 C58LDF 7728944 IC50 > 10000 nM T83875 COS56D 7946925 IC50 = 7560 nM T83875 C0HDR2 8443698 IC50 = 2670 nM T83875 C4P2UQ 8607850 IC50 > 100000 nM T83875 CSW24U 8744495 IC50 > 100000 nM T83875 C95JLG 9412345 IC50 > 100000 nM T83875 C18OMT 9413726 IC50 > 100000 nM T83875 CQ8IR0 9593639 IC50 = 1830 nM T83875 CB41FJ 9601017 IC50 > 10000 nM T83875 C8I7XN 9609596 IC50 = 1790 nM T83875 CF4A5O 9637488 IC50 = 3380 nM T83875 CUFX46 9685369 IC50 = 2040 nM T83875 C79LKI 9737735 IC50 = 16600 nM T83875 CB9IF4 9737737 IC50 = 21300 nM T83875 CV7W8X 9737770 IC50 = 38610 nM T83875 CVSU04 9817917 IC50 > 100000 nM T83875 C03JZN 9838864 IC50 > 50000 nM T83875 CW86OS 9841004 Ki = 2900 nM T83875 C9Z1XQ 9879646 Ki = 58000 nM T83875 CG12HW 9881447 IC50 = 3240 nM T83875 C5BES3 9882402 Ki = 12.6 nM T83875 CFRO05 9904206 Ki = 4.3 nM T83875 C8LR4G 9944468 Ki = 146000 nM T83875 CI19EX 9950622 Ki = 22600 nM T83875 CVY48J 9979525 Ki > 200000 nM T83875 CYO48N 9995644 IC50 = 23988.33 nM T83875 CMZ65T 10025920 Ki = 102000 nM T83875 CW9T3A 10064939 IC50 = 15135.61 nM T83875 C7IEF9 10095474 IC50 = 8930 nM T83875 CRLY52 10126362 Ki = 293000 nM T83875 C3JCQ8 10128237 Ki > 200000 nM T83875 C90EUM 10130534 IC50 = 21000 nM T83875 CE64YJ 10151082 Ki = 47000 nM T83875 CM5FH8 10151157 Ki = 3000 nM T83875 C63PBT 10173120 Ki = 500 nM T83875 CX7ML8 10175195 Ki > 100000 nM T83875 C62ZIW 10176672 IC50 = 11000 nM T83875 CJ4DX0 10193371 Ki = 63000 nM T83875 CSC5F2 10194547 Ki > 200000 nM T83875 C1VR0G 10194605 Ki = 3200 nM T83875 CWQ4V6 10195468 Ki = 16000 nM T83875 CN5F1H 10216656 Ki > 200000 nM T83875 C3PEH7 10246762 IC50 = 3852 nM T83875 CT5Y8O 10309027 Ki = 105000 nM T83875 CXOV50 10312499 Ki > 100000 nM T83875 CD7H4C 10314028 Ki ~ 100000 nM T83875 C65QLI 10331501 IC50 = 13150 nM T83875 CC58YU 10331851 IC50 = 11900 nM T83875 CZ1NI7 10339427 IC50 = 10.7 nM T83875 C1TOA6 10360889 IC50 = 38 nM T83875 CRF71V 10376837 IC50 = 1680 nM T83875 CU5I8C 10379207 IC50 = 41230 nM T83875 C25WON 10382902 IC50 = 20000 nM T83875 CW38VN 10431444 Ki = 25000 nM T83875 C8MA6I 10442609 IC50 = 17100 nM T83875 CIM09T 10443747 IC50 = 4500 nM T83875 CG9Z3B 10470997 IC50 = 123 nM T83875 CR9SE7 10540319 IC50 = 4950 nM T83875 CDT28L 10586897 IC50 = 3300 nM T83875 CA51UC 10633774 IC50 = 38150 nM T83875 CAC7U5 10666499 IC50 = 20140 nM T83875 CFA2E3 10682241 IC50 = 792 nM T83875 C8YO4I 10682287 Ki = 1100 nM T83875 CYV29T 10682625 IC50 = 5140 nM T83875 CW67NI 10705194 IC50 = 1190 nM T83875 C0OW2P 10850658 IC50 = 37730 nM T83875 C79PFH 10855817 IC50 = 71380 nM T83875 C7RD3K 10872091 IC50 > 10000 nM T83875 C3EHA8 10879393 IC50 = 18200 nM T83875 CU4FD9 10883954 Ki = 170 nM T83875 CFL57V 10889774 Ki = 590201080.2 nM T83875 C31MCX 10911003 Ki = 399944749.8 nM T83875 C7DO5I 10921069 IC50 = 7500 nM T83875 CLK8M1 10970782 IC50 > 10000 nM T83875 CPH2B5 10981956 Ki = 290 nM T83875 CM89FA 10987728 Ki = 339625272.6 nM T83875 C8NS7W 11008446 IC50 = 23400 nM T83875 C5OA1U 11055762 IC50 = 396 nM T83875 C7QN1X 11064199 Ki = 539510622.5 nM T83875 CF9K8Z 11064689 Ki = 359749335.2 nM T83875 CTOC87 11077623 IC50 > 100000 nM T83875 C1X3HZ 11085643 Ki = 399944749.8 nM T83875 CX5F2M 11127444 Ki = 500034535 nM T83875 C4YX6G 11127627 Ki = 260015956.3 nM T83875 CL09KJ 11128161 Ki = 199986187 nM T83875 C74VIX 11167787 Ki = 3500 nM T83875 CQY25S 11205968 IC50 = 320000 nM T83875 CRC94Z 11217911 IC50 = 6700 nM T83875 CKEG43 11217912 IC50 = 230000 nM T83875 CU9RL6 11219387 Ki = 3499451.67 nM T83875 CVR53M 11276756 IC50 = 9020 nM T83875 C9Q4IK 11288016 IC50 = 280 nM T83875 C8DK6A 11335051 Ki = 10000000 nM T83875 CLF08H 11355798 IC50 > 100000 nM T83875 C0EG5H 11361757 Ki = 4500 nM T83875 CI9ST4 11382228 IC50 = 11220.18 nM T83875 C6O4QN 11407219 Ki = 1600 nM T83875 CKNY71 11414870 Ki = 100000000 nM T83875 CX6J4S 11420409 Ki > 200000 nM T83875 CN6M2D 11425653 Ki = 9506047.94 nM T83875 C8VJ1K 11481147 IC50 = 40200 nM T83875 C5MOH8 11506668 IC50 = 6000 nM T83875 C2BV6C 11508380 IC50 > 100000 nM T83875 C0KR4I 11510480 Ki > 178000 nM T83875 C2W9XM 11515943 IC50 = 0.1 nM T83875 C6OWB1 11529960 IC50 = 9670 nM T83875 C0FWJ4 11544612 IC50 = 11430 nM T83875 C03FJS 11580776 IC50 > 100000 nM T83875 CP15LR 11597959 Ki = 94000 nM T83875 CKHB97 11603378 Ki = 4300 nM T83875 CXU5I3 11616886 Ki = 15700 nM T83875 CG57SF 11632704 Ki = 48000 nM T83875 C2D7FW 11644221 IC50 = 1000 nM T83875 C6O9WD 11658488 IC50 = 2800 nM T83875 C15VWK 11661838 Ki > 178000 nM T83875 CFUQ76 11668415 Ki = 6000 nM T83875 CS28CV 11674943 IC50 = 16040 nM T83875 C7E9FY 11687666 IC50 = 54650 nM T83875 CD57XZ 11695291 IC50 = 14760 nM T83875 CI18UY 11701511 IC50 = 21740 nM T83875 C3WY1J 11702056 IC50 > 10000 nM T83875 CO3U4B 11705008 Ki > 12000 nM T83875 CV9R5X 11715359 IC50 = 2000 nM T83875 CQ9JE1 11716117 IC50 > 100000 nM T83875 C09YMZ 11746926 Ki = 979489985.4 nM T83875 C82ZEG 11806071 Ki = 149968483.6 nM T83875 CP0FG5 11806940 Ki = 179887091.5 nM T83875 CZV16C 11953368 IC50 = 58000 nM T83875 C4ATG6 12070966 IC50 = 1230 nM T83875 C6KB9J 12070967 IC50 = 13 nM T83875 CMW6C0 12142409 Ki = 16400 nM T83875 C2UYL7 12147097 IC50 > 100000 nM T83875 CM13FC 12200770 IC50 > 100000 nM T83875 C05MGK 12302475 Ki = 2000 nM T83875 CO0B3Y 12317147 Ki = 130000 nM T83875 CQ17RI 12320038 IC50 = 20200 nM T83875 CET0B9 12536095 IC50 > 100000 nM T83875 CN1I4H 12615313 IC50 = 8030 nM T83875 CL19DT 12622120 IC50 > 100000 nM T83875 C01ZKC 12743534 IC50 = 36900 nM T83875 C9BKA2 12822089 IC50 = 16700 nM T83875 CL12FG 12887493 IC50 = 6810 nM T83875 C3HIS0 12899541 IC50 = 6600 nM T83875 CO3FX6 13004209 IC50 = 7530 nM T83875 CW31OY 13067328 IC50 = 238 nM T83875 CX1I4T 13067331 IC50 = 1320 nM T83875 CFJW72 13108121 IC50 = 1100 nM T83875 C9RH7B 13108122 IC50 = 13000 nM T83875 CY6W5B 13147660 IC50 = 720 nM T83875 CN8Y5U 13340061 IC50 = 88430 nM T83875 CSY7V3 13560856 Ki = 55000 nM T83875 C9NHV7 13925346 Ki = 9200 nM T83875 CA93TP 14248936 IC50 = 100000 nM T83875 C65XEY 14364356 IC50 = 14 nM T83875 C8R0DB 14364358 IC50 = 44 nM T83875 C2AM4B 14364359 IC50 = 9810 nM T83875 CC0PF9 14493789 IC50 = 55470 nM T83875 CKR3Q8 14504445 Ki = 1000000 nM T83875 C6BXJ3 14521594 IC50 = 25140 nM T83875 CL8CJ0 14570343 IC50 > 10000 nM T83875 CNWR24 14630571 IC50 = 37000 nM T83875 CHS1K3 14669096 IC50 = 8120 nM T83875 C3H1UG 14737145 IC50 = 40200 nM T83875 CBZ43L 14807789 IC50 = 4600 nM T83875 CEH9F5 14807793 IC50 > 50000 nM T83875 CJZ87V 14810157 Ki = 148 nM T83875 C8ND3J 14920129 IC50 = 80300 nM T83875 C2J8SV 14956421 Ki = 805 nM T83875 C2GJQ3 14956422 Ki = 333 nM T83875 CCW67A 14956425 IC50 = 68870 nM T83875 CJ3E7T 15125273 IC50 > 100000 nM T83875 CK52YI 15127377 IC50 = 40000 nM T83875 CUA6O8 15193131 IC50 > 100000 nM T83875 C7Y2EW 15193139 IC50 = 100000 nM T83875 CRN2Z1 15206345 IC50 = 15450 nM T83875 CNX0G2 15234950 Ki = 4000 nM T83875 C2YLH1 15304541 IC50 = 21410 nM T83875 CIQ3X9 15304544 IC50 > 200000 nM T83875 CHV17I 15324420 Ki = 980 nM T83875 CAY8U5 15480987 IC50 = 78300 nM T83875 C9A1WR 15484393 IC50 = 11460 nM T83875 CNEI48 15521042 Ki = 900 nM T83875 CFGD90 15609637 IC50 > 100000 nM T83875 CB36PW 15634400 IC50 = 0.83 nM T83875 C8FSV7 15953790 IC50 = 37 nM T83875 CJV02O 15953792 IC50 = 299800 nM T83875 C21GMP 16099924 Ki = 1220 nM T83875 CIZ1J8 16110287 Ki = 6998419.96 nM T83875 CHV72Z 16110289 Ki = 39994474.98 nM T83875 CZ1I2G 16110291 Ki = 89949758.15 nM T83875 CHX70R 16110293 Ki = 50003453.5 nM T83875 CVO5A6 16110294 Ki = 50003453.5 nM T83875 CH8U1K 16110295 Ki = 100000000 nM T83875 C7TL0W 16110298 Ki = 260015956.3 nM T83875 C7KAT5 16110299 Ki = 1698243.65 nM T83875 C9XTH8 16110300 Ki = 19998618.7 nM T83875 C3NST4 16110301 Ki = 829850767.5 nM T83875 C0TA1H 16110302 Ki = 439541615.4 nM T83875 CQEP43 16110303 Ki = 330369541 nM T83875 C73CKM 16110304 Ki = 19998618.7 nM T83875 CZU6D2 16368147 IC50 = 207000 nM T83875 C40MHI 16444239 IC50 = 37530 nM T83875 C1OP9D 16787761 Ki = 2490 nM T83875 C04JHC 16792980 Ki = 1220 nM T83875 CXM83Z 17163667 IC50 > 10000 nM T83875 C6X9OR 17165093 IC50 > 10000 nM T83875 C6G9JN 17167188 IC50 > 10000 nM T83875 C56GJX 17391147 IC50 = 4740 nM T83875 CGIP10 17391461 IC50 = 2100 nM T83875 CK72SQ 17392369 IC50 > 100000 nM T83875 C2LP8V 17462470 IC50 > 100000 nM T83875 CUTY36 17469896 IC50 = 40900 nM T83875 CHZ0P1 17749832 IC50 > 10000 nM T83875 C0LAC8 17839878 IC50 > 100000 nM T83875 CC54WV 18093825 IC50 = 18000 nM T83875 CBD6Y7 18526002 IC50 = 970 nM T83875 C82MFL 18684838 Ki = 5900 nM T83875 C4SO6A 19132781 IC50 = 1740 nM T83875 CZTM17 19132783 IC50 = 20500 nM T83875 C2Z6VI 19133248 IC50 = 31450 nM T83875 CI5LJ1 19133249 IC50 = 33884.42 nM T83875 C34IVD 19133250 IC50 = 8128.31 nM T83875 CXR71E 19133252 IC50 = 3900 nM T83875 CMGL84 19133253 IC50 = 20892.96 nM T83875 CBZ2J6 19133254 IC50 = 4250 nM T83875 CX9AL2 19133255 IC50 = 15135.61 nM T83875 C26HDA 19133257 IC50 = 5754.4 nM T83875 C9ACO3 19133259 IC50 = 1950 nM T83875 CP98TF 19133260 IC50 = 45457 nM T83875 C68VCD 19167136 IC50 > 100000 nM T83875 CJ0I9K 19203678 IC50 = 88900 nM T83875 CC85YA 19382380 IC50 = 9400 nM T83875 CJ1GF9 19556945 Ki = 5220 nM T83875 C5IQ9M 19612268 IC50 = 31000 nM T83875 CK49IU 19612271 IC50 = 36000 nM T83875 C76DUN 19752124 IC50 = 15135.61 nM T83875 CR2V8K 20331466 Ki = 25 nM T83875 C8B9FO 20438759 IC50 = 300 nM T83875 CEJ36U 20559176 IC50 = 51660 nM T83875 CK27BD 20740795 Ki = 100 nM T83875 C05XEP 21239588 IC50 = 60490 nM T83875 CJX4A2 21240024 IC50 = 2240 nM T83875 C4EDK3 21671938 IC50 = 2120 nM T83875 CQ81MU 21964538 IC50 = 70500 nM T83875 CTM62N 21974910 Ki = 2500 nM T83875 C5VJ4X 21982105 IC50 = 4160 nM T83875 C2K4WS 22011729 IC50 = 1380 nM T83875 C5YSK9 22055258 IC50 > 100000 nM T83875 CTC8J6 22215549 IC50 > 50000 nM T83875 CZ7L3Q 22421276 IC50 > 100000 nM T83875 CJNT68 22569785 IC50 = 37800 nM T83875 C81HXB 23372523 IC50 > 100000 nM T83875 CYOH73 23454034 IC50 = 13100 nM T83875 CS23FB 23624703 Ki = 5900 nM T83875 C0EGO8 23624706 Ki = 136000 nM T83875 CQ29HW 23626128 Ki < 300 nM T83875 CD9NO4 23626130 Ki = 58000 nM T83875 C0HA4Y 23626131 Ki > 5600 nM T83875 C3Z6LM 23626132 Ki > 89000 nM T83875 CQ9KE5 23626281 Ki > 44000 nM T83875 CWX78R 23626282 Ki = 10500 nM T83875 CHR2L8 23626283 Ki = 15000 nM T83875 C94WCT 23626284 Ki = 28000 nM T83875 C04KXI 23626285 Ki > 44000 nM T83875 C78MWR 23626435 Ki = 1700 nM T83875 C4U0OG 23626436 Ki = 3000 nM T83875 CBMZ61 23626437 Ki = 2500 nM T83875 C28NFE 23626438 Ki = 11300 nM T83875 C2EXB1 23626439 Ki = 4800 nM T83875 CKM12C 23626771 Ki = 700 nM T83875 COI84Z 23626923 Ki > 11000 nM T83875 C7EK4A 23626924 Ki = 19000 nM T83875 C3VCB0 23626925 Ki = 41000 nM T83875 CS9BR5 23626927 Ki = 4500 nM T83875 CS5E6J 23729988 Ki = 546000 nM T83875 C9U0WO 23729989 Ki = 355000 nM T83875 C9Y2EC 23879759 IC50 = 424 nM T83875 C21XUN 23996002 IC50 = 2130 nM T83875 CSJ2B6 24164753 IC50 = 7590 nM T83875 C9R1PK 24180717 IC50 = 23000 nM T83875 C5PG7Y 24230625 IC50 = 31800 nM T83875 C58IBL 24395421 IC50 = 36200 nM T83875 CR1L8S 24397125 IC50 = 184000 nM T83875 CBXC05 24424330 IC50 = 40 nM T83875 CX98YL 24506542 IC50 = 15000 nM T83875 CQZ20A 24506553 IC50 = 1950 nM T83875 CTGB25 24695698 IC50 = 51300 nM T83875 CM2J7N 24799761 IC50 = 147000 nM T83875 C6BUH8 24893999 IC50 = 130 nM T83875 C80WUR 24894016 IC50 = 430 nM T83875 CXRN67 25027416 IC50 = 4760 nM T83875 C6ERN5 25027417 IC50 = 8340 nM T83875 C9PY4E 25027421 IC50 = 190 nM T83875 C9K0YJ 25034467 IC50 = 4940 nM T83875 CH0M8Q 25034468 IC50 = 3530 nM T83875 C97SXU 25034469 IC50 = 4810 nM T83875 C5GAV4 25034470 IC50 = 6830 nM T83875 CVNZ40 25034471 IC50 = 42310 nM T83875 C0I8EP 25034472 IC50 = 43950 nM T83875 CASW39 25034473 IC50 = 7220 nM T83875 CN6DF9 25034474 IC50 = 5495.41 nM T83875 CDVA38 25045938 IC50 = 177500 nM T83875 C4MYE1 25139468 IC50 = 695 nM T83875 CANL42 25139470 IC50 = 255000 nM T83875 CA38ZR 25139472 IC50 = 7.16 nM T83875 C5G4MN 25139474 IC50 = 32800 nM T83875 CC7SL1 25147674 Ki = 920449.57 nM T83875 CTKW89 25147675 Ki = 43954161.54 nM T83875 C8HSP4 25184392 IC50 > 100 ug.mL-1 T83875 C9CT6N 25184393 IC50 = 56.9 ug.mL-1 T83875 CO25XG 25184460 IC50 = 24.4 ug.mL-1 T83875 C3UB2H 25184466 IC50 > 100 ug.mL-1 T83875 CI2GX7 25193423 IC50 = 1047.13 nM T83875 C7VG9E 25193523 IC50 = 2911 nM T83875 CD1YG4 25193524 IC50 = 35220 nM T83875 CD04UK 25193525 IC50 = 23120 nM T83875 C5B7XI 25193526 IC50 = 22760 nM T83875 CNW97L 25193527 IC50 = 3890.45 nM T83875 CJP69X 25193530 IC50 = 7160 nM T83875 CS10DN 25193635 IC50 = 7585.78 nM T83875 C93CIO 25193636 IC50 = 2760 nM T83875 C54USH 25193637 IC50 = 5770 nM T83875 CF69VX 25193638 IC50 = 4260 nM T83875 C63AJF 25193733 IC50 = 6165.95 nM T83875 CP4LK1 25221889 IC50 = 35 nM T83875 CL23IW 25254728 IC50 > 20000 nM T83875 C92TFZ 25335287 IC50 > 500000 nM T83875 CSC9F8 25501843 IC50 > 500000 nM T83875 CRK3Y8 25769005 IC50 > 50000 nM T83875 CP5UF4 25844460 IC50 > 200000 nM T83875 C1CK8A 26216970 IC50 > 100000 nM T83875 C5GRW1 26564219 IC50 > 100000 nM T83875 C0KCL1 28369336 IC50 = 46800 nM T83875 CLZ8F5 28739530 IC50 = 65230 nM T83875 CR6A9X 38763705 IC50 = 13500 nM T83875 CE0G5M 38770453 IC50 = 27200 nM T83875 CU04HR 39082892 Ki = 19100 nM T83875 CRH7M4 39247144 Ki = 190 nM T83875 CFYI84 42601491 IC50 > 30000 nM T83875 C0VQH4 42618005 IC50 = 9330 nM T83875 C7VKO3 42618006 IC50 = 12760 nM T83875 CFR5X6 42618008 IC50 = 63520 nM T83875 C7V8UM 42618009 IC50 = 58640 nM T83875 CG8AX1 42618010 IC50 = 60930 nM T83875 CCW65K 42618011 IC50 = 61380 nM T83875 C58OWA 42618012 IC50 = 51890 nM T83875 C45TRB 42618013 IC50 = 49750 nM T83875 CP2QK3 42618015 IC50 = 52890 nM T83875 C8BL6I 42618017 IC50 = 41400 nM T83875 C5VNE8 42618018 IC50 = 58490 nM T83875 C03VDN 42618019 IC50 = 55830 nM T83875 C19ICQ 42618020 IC50 = 59560 nM T83875 CGE5Q6 42618021 IC50 = 49200 nM T83875 CN38VU 42618022 IC50 = 52620 nM T83875 C3N1XH 42618025 IC50 = 48950 nM T83875 C8EK3R 42623200 IC50 > 30000 nM T83875 CJ4MD2 42623269 IC50 > 30000 nM T83875 CCAW14 42623272 IC50 > 30000 nM T83875 C5N7SE 42624010 IC50 > 30000 nM T83875 CXU9W0 42624092 IC50 > 30000 nM T83875 C7SE6I 42624095 IC50 > 30000 nM T83875 CZ0T8M 42624097 IC50 > 10000 nM T83875 CJR34E 43090939 IC50 = 8520 nM T83875 CDV3A8 43835789 IC50 = 6630 nM T83875 CD0N4Z 44178231 IC50 > 100000 nM T83875 CWR6S9 44205192 Ki = 4000 nM T83875 COI86D 44221695 IC50 = 6571 nM T83875 CWRU07 44269497 Ki = 28.4 nM T83875 CO3RN2 44284812 Ki = 10000 nM T83875 CDJC64 44362531 IC50 = 90400 nM T83875 C52LPH 44371758 IC50 = 1360 nM T83875 C9LZ3A 44371762 IC50 = 13600 nM T83875 CS6Y9L 44371770 IC50 = 650 nM T83875 C9S8PR 44371772 IC50 > 1000000 nM T83875 CW2O7E 44371784 IC50 = 25400 nM T83875 COX76Y 44371839 IC50 = 100 nM T83875 CX1TC7 44371843 IC50 = 920 nM T83875 C2TI1K 44371844 IC50 = 30800 nM T83875 CNZ59L 44371845 IC50 = 113000 nM T83875 C5S4VL 44371849 IC50 = 2120 nM T83875 CB6L5H 44371855 IC50 = 210 nM T83875 C7X0ZU 44371902 IC50 = 540 nM T83875 C81QMK 44371903 IC50 = 750 nM T83875 CYPL76 44371904 IC50 = 5470 nM T83875 CFQ15B 44371906 IC50 = 1610 nM T83875 CY5E0V 44371918 IC50 = 22500 nM T83875 CI25TC 44371926 IC50 = 3740 nM T83875 CPZ38Y 44372077 IC50 > 1000000 nM T83875 C1K8SH 44372226 Ki = 170000 nM T83875 CV9Y3R 44388098 Ki = 3400 nM T83875 C0IH8V 44395951 IC50 = 23000 nM T83875 CJ3F4D 44395980 IC50 = 24000 nM T83875 CT6Y1Z 44396044 IC50 = 18000 nM T83875 CX2D1K 44396070 IC50 = 3300 nM T83875 C6E0ON 44396084 IC50 = 14900 nM T83875 CVN2C1 44396085 IC50 = 37000 nM T83875 CJ0V8I 44396106 IC50 = 27000 nM T83875 CYTW05 44418972 IC50 = 41230 nM T83875 CP4T6L 44430620 Ki = 420 nM T83875 C67ZNA 44437460 IC50 > 10000 nM T83875 C6PK0B 44442374 IC50 = 1995.26 nM T83875 CQ16OE 44442375 IC50 = 3460 nM T83875 CSX23C 44442379 IC50 = 2760 nM T83875 CI1XD0 44448000 IC50 = 375000 nM T83875 CMI7C5 44448037 IC50 = 2390 nM T83875 CT5J2O 44562977 IC50 = 63530 nM T83875 CIL0J4 44562978 IC50 = 2660 nM T83875 CB2F3Y 44563021 IC50 = 20350 nM T83875 CEGS18 44563022 IC50 = 121 nM T83875 C6DFK9 44563083 IC50 = 57920 nM T83875 C59WQS 44565882 IC50 = 25300 nM T83875 CJ8ZA4 44572695 IC50 = 5700 nM T83875 CV21MX 44577626 IC50 = 800 nM T83875 CB1V4I 44577717 IC50 = 76000 nM T83875 CL2TP4 44577718 IC50 = 14000 nM T83875 CT9GO4 44577748 IC50 = 47000 nM T83875 CQ16OW 44582853 IC50 = 7410 nM T83875 C47EYV 44587515 IC50 = 43550 nM T83875 CT9VY0 44587516 IC50 = 44700 nM T83875 C2WV6H 44587534 IC50 = 37950 nM T83875 CWR84V 44587536 IC50 = 31030 nM T83875 CRNH87 44588040 Ki = 5997910.76 nM T83875 C62TQU 44588102 Ki = 3999447.5 nM T83875 CUN1E8 44588103 Ki = 6501296.9 nM T83875 CUL39M 44588104 Ki = 100000000 nM T83875 COU71J 44588137 Ki = 100000000 nM T83875 C95OMJ 44588138 Ki = 1000000000 nM T83875 C1T9RZ 44588171 Ki = 5997910.76 nM T83875 C2LP8Z 44588173 Ki = 138995263.1 nM T83875 CTL18W 44588175 Ki = 1000000 nM T83875 CH9E3V 44588205 Ki = 6998419.96 nM T83875 CX1Q6Y 44588206 Ki = 72945751.03 nM T83875 CT2HZ4 44588207 Ki = 88920111.79 nM T83875 C9TY5H 44588237 Ki = 769130440.3 nM T83875 C0UG7T 44588238 Ki = 11994993.03 nM T83875 C45AGD 44588239 Ki = 699841996 nM T83875 C39UHD 44588240 Ki = 53951062.25 nM T83875 C0IZ7J 44588241 Ki = 10000000 nM T83875 CIHS73 44588242 Ki = 59979107.63 nM T83875 C3HQ0J 44588268 Ki = 102093948.4 nM T83875 CDMR17 44588269 Ki = 65012969.03 nM T83875 CU6S7O 44607264 Ki = 230000 nM T83875 COW48M 44665667 IC50 = 1780 nM T83875 C7ZJH9 44886703 IC50 = 1860 nM T83875 C0P8RX 45113793 IC50 = 50140 nM T83875 C5YKT8 45113794 IC50 = 65840 nM T83875 CB8ZS5 45113924 IC50 = 69450 nM T83875 CM19RV 45113925 IC50 = 69970 nM T83875 CNL38T 45490311 IC50 = 1840 nM T83875 CR8T0C 45490312 IC50 = 11100 nM T83875 C4EN8L 46222450 IC50 > 150000 nM T83875 CI0U9V 46223339 IC50 = 2700 nM T83875 C1JEG9 46236753 IC50 = 24 nM T83875 C09EFO 46467419 Ki = 174630 nM T83875 C6JUK7 46830228 IC50 = 320 nM T83875 C1FN3T 46830229 Ki = 1200 nM T83875 C72IST 46830246 IC50 = 31 nM T83875 CS6W7J 46889939 IC50 = 37000 nM T83875 C4DTN2 46911175 IC50 = 2400 nM T83875 CI7TL1 46944671 Ki = 5470 nM T83875 C8WH1R 46944673 Ki = 3050 nM T83875 C2FT5S 46944674 Ki = 2020 nM T83875 CO7A5T 46944675 Ki = 3290 nM T83875 C63XJZ 46944676 Ki = 1030 nM T83875 C3I8WN 46945877 IC50 = 82 nM T83875 CG58TS 46945878 IC50 = 6.1 nM T83875 CT3IQ0 46945880 IC50 = 87 nM T83875 CE95LB 46945881 IC50 = 6.8 nM T83875 CKD6L8 46946079 IC50 = 2.7 nM T83875 CN7DA6 46946080 IC50 = 88 nM T83875 CV08XW 46946081 IC50 = 6.2 nM T83875 CEFW62 46946082 IC50 = 2.7 nM T83875 C0VLP8 46946083 IC50 = 22 nM T83875 CUFK84 46946084 IC50 = 750 nM T83875 CA80DH 46946273 IC50 = 9.6 nM T83875 CU8G7X 46947641 Ki = 2020 nM T83875 C3OK9X 46947642 Ki = 68270 nM T83875 C1CAN0 46949549 IC50 = 1140 nM T83875 C5E6XN 47002592 IC50 > 30000 nM T83875 C9HW8B 47003377 IC50 > 100000 nM T83875 CC81EY 47398190 IC50 = 12400 nM T83875 CJ29HG 47420565 IC50 = 50600 nM T83875 C3DK8H 49098177 IC50 = 16100 nM T83875 CA6SL4 49863576 IC50 = 1450 nM T83875 C87CZL 49863577 IC50 = 836.21 nM T83875 CG5L1Q 49863578 IC50 = 591.8 nM T83875 CU54BX 49863607 IC50 = 1910 nM T83875 CJW3D5 49863635 IC50 = 737.4 nM T83875 C9TL2A 49863636 IC50 = 678.75 nM T83875 CF9TR0 49863637 IC50 = 749.15 nM T83875 COR75I 49863638 IC50 = 1780 nM T83875 CVX08W 49863730 IC50 = 5560 nM T83875 C52UHN 49864177 Ki = 250000 nM T83875 CPO5C2 49864508 IC50 = 31200 nM T83875 C35XSM 49868483 Ki = 110000 nM T83875 CU5XE6 50745004 IC50 > 100000 nM T83875 CO35KG 50876171 IC50 = 1980 nM T83875 C2X9QA 50876174 IC50 = 1737.8 nM T83875 C7ZPY5 50994008 Ki = 3.6 nM T83875 CS96UB 50994176 Ki = 577 nM T83875 C35DLK 51049245 IC50 > 100000 nM T83875 C4Q6RF 52174704 IC50 = 38400 nM T83875 C38DBE 52446186 IC50 > 100000 nM T83875 C2DBZ5 52541425 IC50 = 83700 nM T83875 CFYQ13 52915138 IC50 = 9670 nM T83875 C0FTO3 52936300 IC50 = 1440 nM T83875 C8TRH1 52940770 IC50 = 4786.3 nM T83875 CVY9C7 52940812 IC50 = 20570 nM T83875 C7NUM5 52941235 IC50 = 59280 nM T83875 C81FZE 52941812 IC50 = 37840 nM T83875 CO42IY 52942005 IC50 = 43550 nM T83875 CO6R7T 52942020 IC50 = 37520 nM T83875 C14CJD 52942390 IC50 = 4436 nM T83875 C09WXG 52942474 IC50 = 9549.93 nM T83875 C0J2FL 52943064 IC50 = 830 nM T83875 C0CB3Z 52943176 IC50 = 6830 nM T83875 CW86YM 52943217 IC50 = 40570 nM T83875 CX0Y2K 52943218 IC50 = 42660 nM T83875 C0HVJ6 52943230 IC50 = 31030 nM T83875 CP5NZ8 52943354 IC50 = 45708.82 nM T83875 CL94WN 52943606 IC50 = 2290.87 nM T83875 C7R0ZB 52944251 IC50 = 50720 nM T83875 CJKO37 52944406 IC50 = 43651.58 nM T83875 C98VBM 52945642 IC50 = 3530 nM T83875 CD40XF 52945645 IC50 = 4940 nM T83875 CI9Y4H 52945649 IC50 = 10090 nM T83875 C6JKN7 52945917 IC50 = 19498.45 nM T83875 CBD1G2 52946045 IC50 = 7079.46 nM T83875 CD85UQ 52946066 IC50 = 10279 nM T83875 CJX6E9 52946067 IC50 = 7229 nM T83875 CP51KJ 52946520 IC50 = 42310 nM T83875 CJ7SQ1 52946862 IC50 = 38840 nM T83875 C5NQ0L 52946864 IC50 = 21900 nM T83875 C2EQ0Z 52947352 IC50 = 4327 nM T83875 CO0D3Z 52947695 IC50 = 23988.33 nM T83875 CG9X5N 52948086 IC50 = 5500 nM T83875 CZIW51 52948923 IC50 = 40320 nM T83875 CM2H4L 52949147 IC50 = 19620 nM T83875 C12DYG 52949244 IC50 = 37950 nM T83875 CKE8D5 52949315 IC50 = 35220 nM T83875 CM9B7Z 52949317 IC50 = 44700 nM T83875 C89GLO 52949320 IC50 = 43780 nM T83875 CS32GV 52949324 IC50 = 17140 nM T83875 CS9NO2 52949516 IC50 = 4786.3 nM T83875 CJC20G 52949550 IC50 = 81283.05 nM T83875 CK15PD 52950170 IC50 = 7220 nM T83875 CGQ76K 53009757 IC50 = 61400 nM T83875 CVZ2D4 53248704 IC50 = 20740 nM T83875 C6Z0BI 53315284 IC50 = 11500 nM T83875 C7AT0L 53316832 Ki = 24.9 nM T83875 CP39IR 53317196 Ki = 3210 nM T83875 C16VWZ 53318151 Ki = 29.5 nM T83875 CU13PW 53318152 Ki = 100 nM T83875 C5B6IR 53319012 Ki = 255.7 nM T83875 CG7R9F 53319492 Ki = 3.9 nM T83875 C9UD2P 53319928 Ki = 1290 nM T83875 C27VRY 53322102 Ki = 5 nM T83875 CS0F1P 53322103 Ki = 5 nM T83875 C0F5JO 53322104 Ki = 35.4 nM T83875 CKZ0C3 53322381 IC50 > 100000 nM T83875 CW81FC 53322432 Ki = 1830 nM T83875 C2MO5K 53324249 Ki = 1023.8 nM T83875 C8XZ6A 53326058 Ki = 684 nM T83875 C6M8PN 53326896 Ki = 500 nM T83875 C76GDP 53358665 Ki = 7000 nM T83875 CIVP93 53361170 IC50 = 20350 nM T83875 C5BM2I 53361171 Ki = 5310 nM T83875 CQ2Z4F 53361172 Ki = 580 nM T83875 CUI4C7 53361173 Ki = 460 nM T83875 C19YQZ 53361174 Ki = 470 nM T83875 C6Z0DN 53375709 Ki = 4810 nM T83875 C7PNY9 53375710 Ki = 7980 nM T83875 CHNB31 53375711 Ki = 58710 nM T83875 C89TBV 53375712 Ki = 640 nM T83875 C7TM8P 53387408 IC50 = 11110 nM T83875 CKCG05 53392601 IC50 = 1080 nM T83875 CKH85U 53484089 Ki = 58 nM T83875 CY3F4K 53484090 Ki = 285 nM T83875 C5VKC4 53484091 Ki = 200 nM T83875 CPKR28 53484109 Ki = 285 nM T83875 C0VD5I 54327402 IC50 = 86100 nM T83875 C5I7JA 54526203 IC50 = 3770 nM T83875 CH46TC 54580417 Ki = 82035154.43 nM T83875 CUI7H8 54586284 Ki = 76032627.69 nM T83875 C6D9IE 54753443 IC50 = 47300 nM T83875 CR61HF 54753444 IC50 = 35600 nM T83875 CAG3F4 55285162 IC50 = 170 nM T83875 CIGK63 55471034 IC50 = 20300 nM T83875 CYC5V0 55471035 IC50 = 129000 nM T83875 C5R1CX 56594088 IC50 = 24900 nM T83875 CI8F9G 56594236 IC50 = 35040 nM T83875 C54NUW 56594237 IC50 = 21580 nM T83875 CBX47T 56603017 IC50 = 161 nM T83875 CGA7P8 56640831 IC50 = 39560 nM T83875 C6PSX2 56640832 IC50 = 58430 nM T83875 CU1T2L 56640833 IC50 = 48020 nM T83875 CJ8O3M 56640990 IC50 = 335000 nM T83875 C93UAM 56640991 IC50 = 98200 nM T83875 C5X8JV 56640992 IC50 = 105000 nM T83875 CD0ST5 56640993 IC50 = 74800 nM T83875 C0JXD8 56640994 IC50 = 58400 nM T83875 CDU32V 56640995 IC50 = 34500 nM T83875 CMVU62 56642649 IC50 = 55160 nM T83875 CQL3T5 56642783 IC50 = 46350 nM T83875 CO6QD8 56658693 IC50 = 50510 nM T83875 CK0SB8 56659353 Ki = 940 nM T83875 CE2BN7 56659354 Ki = 2370 nM T83875 C2N1XU 56659718 Ki = 250 nM T83875 CN7W5K 56659719 Ki = 490 nM T83875 CP36XA 56662172 IC50 = 26230 nM T83875 C5WM4L 56663182 Ki = 90 nM T83875 CVP6U5 56665630 IC50 = 380100 nM T83875 CFL96D 56668520 IC50 = 37260 nM T83875 C9EX4Z 56670040 Ki = 360 nM T83875 C24DGB 56670041 Ki = 300 nM T83875 CTM1D9 56670052 IC50 = 46810 nM T83875 CA50XS 56670279 IC50 = 40470 nM T83875 CD84RE 56670280 IC50 = 40550 nM T83875 C6CN3P 56673197 Ki = 460 nM T83875 CZQ8I0 56673343 Ki = 350 nM T83875 CR4BD5 56673554 Ki = 300 nM T83875 CU7FR3 56673555 Ki = 310 nM T83875 CVRQ94 56673556 Ki = 670 nM T83875 CJ8GY0 56673572 IC50 = 19170 nM T83875 CUD04Q 56676876 Ki = 100 nM T83875 CBX28Q 56676877 Ki = 130 nM T83875 C3UEL1 56680195 Ki = 2150 nM T83875 C2LV9D 56683530 Ki = 310 nM T83875 CC8A4B 56683531 Ki = 456 nM T83875 CH1LS7 56683532 Ki = 400 nM T83875 CEML01 56683533 Ki = 150 nM T83875 COLW37 56709688 IC50 > 100000 nM T83875 CXI01A 56807126 IC50 = 21100 nM T83875 CL16UQ 56949326 IC50 < 10000 nM T83875 C0VI8M 56950927 IC50 = 2620 nM T83875 C81FBW 56966263 IC50 = 1720 nM T83875 CXD3C0 57303200 IC50 = 5840 nM T83875 CRF07B 57325839 IC50 = 26700 nM T83875 C4RG0D 57328315 IC50 = 2300 nM T83875 C8TN7H 57335751 IC50 = 38700 nM T83875 CN28HO 57340730 IC50 = 399 nM T83875 C7L2FP 57340731 IC50 = 6.6 nM T83875 CE6LJ1 57379747 IC50 = 3120 nM T83875 CJ12FR 57379748 IC50 = 1910 nM T83875 CVW96L 57379749 IC50 = 424 nM T83875 C60GZY 57379750 IC50 = 106 nM T83875 CCED62 57379751 IC50 = 386 nM T83875 C28HTP 57379977 IC50 = 95 nM T83875 CM72YD 57379978 IC50 = 1230 nM T83875 CAE03J 57379979 IC50 = 322 nM T83875 CG43VX 57379980 IC50 = 1130 nM T83875 C16SCD 57379981 IC50 = 3490 nM T83875 CN0L3H 57379982 IC50 = 255 nM T83875 COX83F 57379983 IC50 = 175 nM T83875 C94HLT 57379984 IC50 = 879 nM T83875 CCD0W7 57380218 IC50 = 480 nM T83875 CQW5T3 57387397 IC50 = 3520 nM T83875 CGSX75 57392339 IC50 = 18700 nM T83875 C1PJO0 57392340 IC50 = 24400 nM T83875 CZ53IA 57392341 IC50 = 3600 nM T83875 C3XO9E 57392561 IC50 = 31300 nM T83875 C0RUX5 57392562 IC50 = 20400 nM T83875 CRAF46 57392799 IC50 > 2000 nM T83875 C2COB9 57394022 IC50 = 5780 nM T83875 C54XIL 57394023 IC50 = 37700 nM T83875 C0Z7SL 57396037 IC50 = 6550 nM T83875 C3CWN6 57397563 IC50 = 30900 nM T83875 CZ90QM 57397635 IC50 = 15500 nM T83875 CG5N1V 57397741 Ki = 15000 nM T83875 C6A1YR 57397784 IC50 = 12000 nM T83875 CTV5M3 57399451 IC50 = 110800 nM T83875 CC5JQ1 57399500 IC50 = 22700 nM T83875 CL8FQ1 57399501 IC50 = 21200 nM T83875 CIY0U2 57399502 IC50 = 8540 nM T83875 CH47EP 57399503 IC50 = 11300 nM T83875 C9PE1R 57401006 IC50 = 107000 nM T83875 CW9R4F 57401210 IC50 = 27300 nM T83875 CQ1D3R 57401211 IC50 = 6100 nM T83875 C5ZBW3 57401260 IC50 = 3220 nM T83875 CR12SB 57401261 IC50 = 18300 nM T83875 CJ3RM8 57402930 Ki = 16000 nM T83875 C3NP9V 57402959 Ki = 407900 nM T83875 CXH24K 58215717 IC50 > 10000 nM T83875 C78KDY 58215749 IC50 = 210 nM T83875 C2R5US 58495647 IC50 = 9870 nM T83875 C5H6GV 58697749 IC50 = 3.8 ug.mL-1 T83875 C1DER5 59601689 IC50 = 5590 nM T83875 C68XHY 60161811 IC50 > 1000 nM T83875 CD6B5P 60203904 IC50 = 2400 nM T83875 C2WQN8 60264513 IC50 > 100000 nM T83875 COHF58 60264536 IC50 > 100000 nM T83875 C3JYI8 60351355 IC50 = 69400 nM T83875 CJYV91 60373147 IC50 = 51800 nM T83875 CTH3G9 60714993 IC50 > 10000 nM T83875 C3XC5K 60715051 IC50 > 10000 nM T83875 CL9QK4 60715052 IC50 > 10000 nM T83875 C0ID4P 60715244 IC50 > 10000 nM T83875 C3Z4GX 60772162 IC50 = 39270 nM T83875 CCJ0Q9 61242666 IC50 > 10000 nM T83875 C41OAY 61832262 IC50 = 392 nM T83875 CF87MH 61832641 IC50 = 2090 nM T83875 C0L8SP 61832822 IC50 = 1290 nM T83875 CMU52G 61833183 IC50 = 311 nM T83875 CS04ZK 61833537 IC50 = 1160 nM T83875 CN54TI 61833721 IC50 = 656 nM T83875 C7BG9L 61833723 IC50 = 207 nM T83875 CDK32Q 61834439 IC50 = 212 nM T83875 CA7P8O 61834440 IC50 = 24 nM T83875 C0E8MG 63095539 IC50 = 46360 nM T83875 C60JPX 63718419 IC50 = 1300 nM T83875 CL7R0T 63937924 IC50 > 10000 nM T83875 C17WZV 64789040 IC50 > 10000 nM T83875 C4RV3T 65477805 IC50 = 1290 nM T83875 C1A3FG 66523802 IC50 > 10000 nM T83875 CB6CU0 66630014 IC50 > 37500 nM T83875 CO84GD 66712998 IC50 = 1030 nM T83875 C1GXR4 69889948 IC50 = 3700 nM T83875 C3PDQ5 70682249 IC50 = 19700 nM T83875 CYG64Z 70682250 IC50 = 1530 nM T83875 CFYC13 70684340 IC50 = 6460 nM T83875 CI5ZC4 70684852 IC50 = 13200 nM T83875 CY39PE 70684853 IC50 = 10700 nM T83875 CW3TY2 70684854 IC50 = 44700 nM T83875 C7IG3N 70684855 IC50 = 117000 nM T83875 CYS03B 70686497 IC50 = 143000 nM T83875 CYM2D6 70686498 IC50 = 52900 nM T83875 CMW14V 70687001 IC50 = 8220 nM T83875 CJNL16 70688596 IC50 = 2900 nM T83875 CJ32UT 70689077 IC50 = 34000 nM T83875 CYX4M9 70689078 IC50 = 4590 nM T83875 C4G5FW 70689079 IC50 = 18800 nM T83875 CY05LV 70689080 IC50 = 139000 nM T83875 CI1Q2S 70689082 IC50 = 142000 nM T83875 C12QAY 70690656 IC50 = 1040 nM T83875 C6NWQ7 70690657 IC50 = 103000 nM T83875 CCK52V 70691189 IC50 = 20800 nM T83875 CP3V7G 70691190 IC50 = 372000 nM T83875 C0M7EU 70692804 IC50 = 2200 nM T83875 CAT52I 70692805 IC50 = 15800 nM T83875 CIN7O4 70692806 IC50 = 6260 nM T83875 C0RM9W 70693292 IC50 = 21100 nM T83875 CD5T8W 70693293 IC50 = 20400 nM T83875 C9I3PY 70693294 IC50 = 19400 nM T83875 CQ9NO2 70694840 IC50 = 60600 nM T83875 C7VGX8 70695387 IC50 = 23800 nM T83875 CQ4U0F 70695388 IC50 = 50100 nM T83875 CJBL13 70695389 IC50 = 51800 nM T83875 CB7R4L 70695390 IC50 = 41300 nM T83875 C3KFZ2 70695391 IC50 = 31600 nM T83875 CT8E7W 70696891 IC50 = 143000 nM T83875 CNR15V 70697409 IC50 = 66200 nM T83875 CTFG16 70702063 IC50 = 1520 nM T83875 CI69QM 70702068 IC50 = 1170 nM T83875 CXLT46 70702073 IC50 = 1970 nM T83875 C18MPL 70723639 IC50 > 200000 nM T83875 C7L6PQ 70804892 IC50 = 11100 nM T83875 CZT65E 71081197 Ki = 1840 nM T83875 CON49H 71261649 IC50 > 20000 nM T83875 C2DI4G 71351539 IC50 = 3800 nM T83875 C2Q0VE 71419878 IC50 = 25340 nM T83875 C42BYX 71449560 IC50 = 1680 nM T83875 CQ3OZ8 71450450 IC50 = 623 nM T83875 CZ5H9R 71450578 IC50 = 141000 nM T83875 CCW1Z5 71450579 IC50 = 6430 nM T83875 C3FC2B 71450580 IC50 = 108000 nM T83875 C2G1FO 71451363 IC50 = 958 nM T83875 COP81R 71451364 IC50 = 1010 nM T83875 CWHM59 71452280 IC50 = 2100 nM T83875 CLB25C 71452281 IC50 = 7190 nM T83875 C6I2MP 71452416 IC50 = 125000 nM T83875 C7F4XP 71452417 IC50 = 5660 nM T83875 CLE84D 71452418 IC50 = 250000 nM T83875 CK3G4B 71453169 IC50 = 273 nM T83875 C1T8YS 71454081 IC50 = 5960 nM T83875 C1U2GV 71454184 IC50 = 12000 nM T83875 C0CJV9 71454185 IC50 = 203000 nM T83875 CBQ74P 71455816 IC50 = 54300 nM T83875 CJO48H 71455926 IC50 = 168000 nM T83875 CJ4B2W 71456691 IC50 = 1920 nM T83875 CJTE73 71456692 IC50 = 2270 nM T83875 CS5X1P 71457606 IC50 = 54700 nM T83875 C87RFW 71457723 IC50 = 5700 nM T83875 CRL5P4 71457724 IC50 = 48100 nM T83875 CUIF34 71457725 IC50 = 708 nM T83875 C9UHF3 71458533 IC50 = 1630 nM T83875 CBX0C4 71459629 IC50 = 14700 nM T83875 CL0HS2 71459630 IC50 = 239000 nM T83875 C7I2JG 71459631 IC50 = 3530 nM T83875 C8UJ0T 71460379 IC50 = 506 nM T83875 C4N8JG 71461236 IC50 = 218000 nM T83875 C1L7MK 71461237 IC50 = 129000 nM T83875 C7HA0O 71461238 IC50 = 19000 nM T83875 CRPA65 71461239 IC50 = 2780 nM T83875 C1PG9R 71461375 IC50 = 57300 nM T83875 CL1FP5 71461376 IC50 = 8460 nM T83875 C85UCB 71462073 IC50 = 380 nM T83875 C6G4XF 71462972 IC50 = 1450 nM T83875 CG01AM 71508602 IC50 > 2000 nM T83875 CI1C7E 71508637 IC50 > 2000 nM T83875 C36MKD 71508638 IC50 > 2000 nM T83875 CJP68B 71543365 IC50 = 48300 nM T83875 CW2T6C 71559776 IC50 = 172 nM T83875 CVQ8S3 71559777 IC50 = 227 nM T83875 C9UM3S 71559778 IC50 = 542 nM T83875 CJ7O6M 71559779 IC50 = 303 nM T83875 C2DM5F 71559780 IC50 = 344 nM T83875 CMZ38H 71559781 IC50 = 1060 nM T83875 CCXO52 71559911 IC50 = 629 nM T83875 CSD8O4 71559912 IC50 = 3210 nM T83875 C73IBL 71559913 IC50 = 498 nM T83875 CKH79U 71559914 IC50 = 1070 nM T83875 C3RP6O 71559915 IC50 = 7330 nM T83875 CEZ32S 71559916 IC50 = 1910 nM T83875 CZS83E 71559917 IC50 = 137 nM T83875 C8NKJ7 71559918 IC50 = 240 nM T83875 CBHX24 71560037 IC50 = 323 nM T83875 CDO3U5 71560038 IC50 = 185 nM T83875 CD9UX7 71560039 IC50 = 59900 nM T83875 C0FJ1X 71561478 IC50 > 10000 nM T83875 CYZE35 71561479 IC50 = 2022 nM T83875 CF4T7N 71561482 IC50 = 2870 nM T83875 C13TRN 71561483 IC50 > 10000 nM T83875 C43UWM 71561593 IC50 > 10000 nM T83875 C2GOS6 71562556 IC50 = 726.3 nM T83875 C1RQ0X 71562925 IC50 = 3110 nM T83875 CJ5M2B 71562926 IC50 > 10000 nM T83875 C3XTO4 71562929 IC50 = 1237 nM T83875 C1SYX5 71563047 IC50 = 5690 nM T83875 CX40FP 71563048 IC50 = 812.3 nM T83875 C2A9VU 71563049 IC50 = 10000 nM T83875 CHVB51 71563050 IC50 > 10000 nM T83875 C4N2XD 71563051 IC50 > 1000 nM T83875 CL60DA 71563052 IC50 = 1300 nM T83875 C41JWM 71563053 IC50 = 1632 nM T83875 C4DE7M 71563176 IC50 > 10000 nM T83875 C5DZM0 71563297 IC50 > 10000 nM T83875 CU6NX9 71568925 IC50 = 15370 nM T83875 CY91WT 71568929 IC50 = 1560 nM T83875 CSYG87 71569082 IC50 = 1030 nM T83875 C26OKQ 71569083 IC50 = 25160 nM T83875 C6S5CK 71569084 IC50 = 1430 nM T83875 CSM4W0 71616357 IC50 > 1250000 nM T83875 CQ3I9J 71616361 IC50 > 1250000 nM T83875 CJTX03 71652416 IC50 = 9050 nM T83875 CK1FR2 71652417 IC50 = 2860 nM T83875 CK57NM 71652418 IC50 = 521.4 nM T83875 CJNR53 71652419 IC50 = 192.6 nM T83875 C5HPG0 71652824 IC50 > 1250000 nM T83875 CA8BI9 71654261 IC50 = 33790 nM T83875 CA73CM 71654421 IC50 = 4860 nM T83875 CM20YQ 71654422 IC50 = 43380 nM T83875 C4Y0SL 71654423 IC50 = 7000 nM T83875 C1TPO4 71654581 IC50 = 1260 nM T83875 C9HL6M 71654582 IC50 = 397.8 nM T83875 C6V1HF 71654583 IC50 = 591 nM T83875 C4D0WN 71654584 IC50 = 372.4 nM T83875 C79DOY 71654585 IC50 = 313 nM T83875 C4EQA2 71717323 IC50 > 100000 nM T83875 C4BVA5 71717928 IC50 > 10000 nM T83875 CG4PR6 71764406 IC50 = 8190 nM T83875 CI4Q6K 71764831 IC50 = 7080 nM T83875 CLC90S 71818857 IC50 = 59500 nM T83875 CP07TK 71818858 IC50 = 28600 nM T83875 CJ6ON9 71818859 IC50 = 30200 nM T83875 C4LW8O 71818860 IC50 = 61600 nM T83875 CB48KD 72164304 IC50 = 2840 nM T83875 C5QO7E 72164305 IC50 = 1820 nM T83875 CE6FJ2 72164306 IC50 = 3000 nM T83875 CXQ0T2 72164307 IC50 = 3260 nM T83875 C4PB7G 72164427 IC50 = 50990 nM T83875 C1REN4 72191056 IC50 = 22500 nM T83875 CN56AJ 72191362 IC50 = 19700 nM T83875 CHE87W 72191363 IC50 > 100000 nM T83875 C3RYV1 72191364 IC50 = 7980 nM T83875 C81BYJ 72191365 IC50 = 53700 nM T83875 CHL70P 72191366 IC50 = 22500 nM T83875 C27CBN 72206251 IC50 = 9900 nM T83875 C3BEM8 72696145 IC50 > 10000 nM T83875 C1E4ZD 72696146 IC50 > 10000 nM T83875 CQ35NL 72696147 IC50 > 10000 nM T83875 CRN4B1 72696148 IC50 > 10000 nM T83875 C0IF1J 72696149 IC50 > 10000 nM T83875 CL2H7Y 72696273 IC50 > 10000 nM T83875 C7MX9Y 72696274 IC50 > 10000 nM T83875 CPI89R 72696276 IC50 > 10000 nM T83875 C1RFY6 72696398 IC50 > 10000 nM T83875 C6A8ZF 72696400 IC50 > 10000 nM T83875 C4DN3V 72696521 IC50 > 10000 nM T83875 C81TXZ 72697651 IC50 > 10000 nM T83875 CA5BI1 72697652 IC50 > 10000 nM T83875 C50SYX 72697785 IC50 > 10000 nM T83875 CXPB58 72697786 IC50 > 10000 nM T83875 CJ5W1R 72697787 IC50 > 10000 nM T83875 CY1I8G 72697789 IC50 > 10000 nM T83875 CCOP98 72698081 IC50 > 10000 nM T83875 C50ZUX 72698082 IC50 > 10000 nM T83875 CZG6V9 72698083 IC50 > 10000 nM T83875 CH6Z2U 72698223 IC50 > 10000 nM T83875 C3QVP5 72698224 IC50 > 10000 nM T83875 CST61L 72698226 IC50 > 10000 nM T83875 CKP9M2 72698228 IC50 > 10000 nM T83875 CHDB60 72793898 IC50 > 200000 nM T83875 C3WZD5 73349093 IC50 = 6910 nM T83875 C1D9XC 73354979 Ki = 4000 nM T83875 C3KGJ6 73356295 Ki = 2000 nM T83875 CPG73S 73417116 IC50 = 240 nM T83875 CGD8R4 73671789 IC50 = 6700 nM T83875 C56INT 75395884 IC50 = 553 nM T83875 C74SVL 75414421 IC50 > 100000 nM T83875 CI9Q0G 76281715 IC50 > 25000 nM T83875 C24XKD 76308234 IC50 = 8600 nM T83875 C68RKH 76310231 IC50 = 8900 nM T83875 CDK4R2 76310423 IC50 = 6320 nM T83875 CR1D2Z 76310442 IC50 = 1950 nM T83875 C3N5VB 76310836 IC50 > 10000 nM T83875 C3XPT4 76310839 IC50 = 2680 nM T83875 C9L3GR 76311136 IC50 = 4400 nM T83875 C5LW4R 76311137 IC50 = 980 nM T83875 C7SX1Z 76311199 IC50 = 29830 nM T83875 CJ1W2I 76311204 IC50 > 100000 nM T83875 CVJW69 76311323 IC50 = 28400 nM T83875 CF4YT3 76311324 IC50 = 132000 nM T83875 C70MNC 76311325 IC50 > 500000 nM T83875 C3N4EY 76311326 IC50 = 29300 nM T83875 CP8L3T 76311327 IC50 = 4810 nM T83875 CL8N5U 76314097 IC50 = 3770 nM T83875 CJSF07 76314454 IC50 = 818 nM T83875 C8ZI4Y 76314455 IC50 = 953 nM T83875 CBKZ86 76314456 IC50 > 10000 nM T83875 CO8G2Y 76314457 IC50 = 77.2 nM T83875 CG70QL 76314458 IC50 > 10000 nM T83875 C59NQU 76314463 IC50 = 62.7 nM T83875 C8FTG6 76314464 IC50 > 10000 nM T83875 C1TFS4 76314802 IC50 = 37460 nM T83875 CM5I9G 76314803 IC50 = 89430 nM T83875 C2A8LT 76314813 IC50 > 100000 nM T83875 CK53JN 76314916 IC50 = 40300 nM T83875 C83COP 76314917 IC50 > 500000 nM T83875 C4TCX5 76314918 IC50 = 11300 nM T83875 C59ZBF 76317227 IC50 > 100000 nM T83875 CTX07R 76317228 IC50 > 100000 nM T83875 CO1EN3 76317452 IC50 = 35400 nM T83875 CV6T1W 76317649 IC50 > 100000 nM T83875 CI9Z6N 76317651 IC50 = 4480 nM T83875 CC0B5D 76318043 IC50 = 9.64 nM T83875 CR45HD 76318044 IC50 > 10000 nM T83875 CVDH35 76318045 IC50 = 66.8 nM T83875 CPB7I3 76318046 IC50 > 10000 nM T83875 CKA48M 76318048 IC50 = 10000 nM T83875 CY2QP8 76318337 IC50 = 5.495 nM T83875 CZ31JI 76318338 IC50 = 1530 nM T83875 CA5K6L 76318339 IC50 > 100000 nM T83875 CM97RB 76318340 IC50 = 4260 nM T83875 C38XFN 76318410 IC50 = 24270 nM T83875 C5JB3L 76318411 IC50 > 100000 nM T83875 CL4PU0 76318412 IC50 > 100000 nM T83875 C53ZLX 76318419 IC50 = 89650 nM T83875 C1C5FO 76318420 IC50 > 100000 nM T83875 C4KLE9 76318530 IC50 > 500000 nM T83875 CC50ZL 76318532 IC50 = 53200 nM T83875 CV9MQ4 76318533 IC50 > 500000 nM T83875 CM54SP 76320939 IC50 > 30000 nM T83875 C6XRT0 76321186 IC50 < 1000 nM T83875 C81DZU 76321374 IC50 = 4240 nM T83875 CSZ69D 76321757 IC50 > 10000 nM T83875 CFD09Y 76321758 IC50 > 10000 nM T83875 CU5NB3 76321759 IC50 > 10000 nM T83875 C0PW1A 76321760 IC50 > 10000 nM T83875 C84HGW 76321761 IC50 > 10000 nM T83875 CA3VD4 76321762 IC50 = 930 nM T83875 CSL45N 76321763 IC50 = 59.9 nM T83875 CC90FV 76322024 IC50 > 100000 nM T83875 CEI0B9 76322086 IC50 > 100000 nM T83875 CT8JY2 76322189 IC50 = 9500 nM T83875 CWCI08 76322190 IC50 = 25800 nM T83875 CTH0U1 76322191 IC50 = 14500 nM T83875 C83GJS 76322192 IC50 > 500000 nM T83875 CVXT29 76324406 Ki = 226000 nM T83875 CNS28Q 76324968 IC50 = 1460 nM T83875 C7VMB2 76324978 IC50 = 2160 nM T83875 CV29DJ 76325379 IC50 > 10000 nM T83875 CLU08E 76325380 IC50 > 10000 nM T83875 C7QV3I 76325640 IC50 > 100000 nM T83875 C0X6JA 76325641 IC50 = 100000 nM T83875 C2F4MQ 76325697 IC50 > 100000 nM T83875 CIT8F0 76325703 IC50 > 100000 nM T83875 CA0X3B 76325809 IC50 = 117900 nM T83875 CU9I8M 76325810 IC50 > 500000 nM T83875 C31JLR 76328918 IC50 > 10000 nM T83875 CW14BN 76328919 IC50 = 367 nM T83875 CSR0P3 76328920 IC50 = 74.8 nM T83875 CERI13 76329220 IC50 > 100000 nM T83875 C0ED6S 76329275 IC50 = 90350 nM T83875 CD0OG4 76329396 IC50 = 89300 nM T83875 CCU16Y 76329397 IC50 = 38300 nM T83875 C0NL9S 76329398 IC50 = 33000 nM T83875 CN34ZA 76329399 IC50 = 49200 nM T83875 CWK86G 76329400 IC50 > 500000 nM T83875 CUY96G 76329401 IC50 > 500000 nM T83875 C3PHJ5 76329402 IC50 = 6500 nM T83875 C5DS0O 76329943 IC50 = 5700 nM T83875 CDM84V 76332211 IC50 = 8460 nM T83875 CI8QE0 76332226 IC50 > 100000 nM T83875 CCR1U2 76332604 IC50 = 10000 nM T83875 CUS43N 76332873 IC50 = 100000 nM T83875 CL4WZ8 76332874 IC50 > 100000 nM T83875 CW20MH 76332875 IC50 > 100000 nM T83875 CAEF41 76332923 IC50 = 17580 nM T83875 C91ENH 76332927 IC50 = 97380 nM T83875 C4PRU7 76332928 IC50 > 100000 nM T83875 CO14DA 76333043 IC50 = 108000 nM T83875 C10HPW 76333045 IC50 > 500000 nM T83875 CXG5C1 76333046 IC50 = 248000 nM T83875 C4I0PD 76333047 IC50 > 500000 nM T83875 CV1P3Z 76333048 IC50 > 500000 nM T83875 CK0SM6 76333049 IC50 > 500000 nM T83875 C3B2GE 76334701 IC50 = 233 nM T83875 C6XD0G 76335238 Ki = 4900 nM T83875 C67EJQ 76335845 IC50 = 17100 nM T83875 C2AEN5 76336201 IC50 > 10000 nM T83875 CN0LI4 76336202 IC50 = 66.1 nM T83875 CG41IF 76336203 IC50 = 1570 nM T83875 CUNV46 76336531 IC50 > 100000 nM T83875 CH2T1L 76336532 IC50 = 33090 nM T83875 CKD2R8 76336533 IC50 > 100000 nM T83875 CD2J6U 76336534 IC50 > 100000 nM T83875 C0EXZ4 76336541 IC50 > 100000 nM T83875 C3TW1I 76336666 IC50 = 25300 nM T83875 C34RKL 76336667 IC50 = 44200 nM T83875 C9U8JP 77844601 IC50 >= 10000 nM T83875 C3OP9Q 77844603 IC50 = 8790 nM T83875 CH5YI4 77844667 IC50 = 0.389 nM T83875 C83HNQ 77844716 IC50 = 1.445 nM T83875 CYS0H9 77844719 IC50 = 562 nM T83875 CL40EH 77844721 IC50 = 764 nM T83875 CU6K3W 77844723 IC50 < 10000 nM T83875 C9H7OG 77844769 IC50 > 10000 nM T83875 CUH8Z1 77844770 IC50 > 10000 nM T83875 C5VZ9M 77844771 IC50 > 10000 nM T83875 CR1Y5G 77844772 IC50 < 10000 nM T83875 C7LDN8 86046220 IC50 > 100000 nM T83875 C46NHO 86298552 IC50 = 1290 nM T83875 C74WUO 86729878 IC50 = 140 nM T83875 CJ64QM 86729882 IC50 = 220 nM T83875 C4YE0G 87057445 IC50 > 1250000 nM T83875 CAE9S6 90197458 IC50 = 6800 nM T83875 C97DGB 90197459 IC50 = 1920 nM T83875 CP4FQ2 90197685 IC50 = 235 nM T83875 CB2RV3 90197737 IC50 = 2590 nM T83875 CJW98L 90197739 IC50 = 3510 nM T83875 C6AK9N 90197969 IC50 = 1430 nM T83875 CS0ZH6 90197974 IC50 = 8310 nM T83875 CN7BV6 90479835 IC50 > 10000 nM T83875 CO51GW 90643508 IC50 = 32440 nM T83875 CB0AP6 90643928 IC50 = 547 nM T83875 C0QA7Z 90645389 IC50 = 22690 nM T83875 CF8T2J 90645390 IC50 = 42310 nM T83875 CG98IK 90645391 IC50 = 10080 nM T83875 CG1N2A 90645392 IC50 = 22690 nM T83875 C15POS 90645393 IC50 = 39740 nM T83875 CD48PL 90645394 IC50 = 48270 nM T83875 C9PIU7 90645500 IC50 = 164000 nM T83875 C8ZGF2 90645501 IC50 = 56800 nM T83875 CA8YH9 90645502 IC50 = 93200 nM T83875 CLJ8O4 90645503 IC50 = 19500 nM T83875 C8QI3X 90645505 IC50 = 86600 nM T83875 CR7UD8 90645506 IC50 = 9930 nM T83875 C03REM 90646727 IC50 > 10000 nM T83875 C8RE0M 90646728 IC50 > 10000 nM T83875 CZF90P 90646729 IC50 > 10000 nM T83875 CV95XQ 90646731 IC50 > 10000 nM T83875 CV6X7K 90646732 IC50 > 10000 nM T83875 C8I7JS 90646833 IC50 > 10000 nM T83875 C40MQW 90656446 IC50 = 13060 nM T83875 CF5I3K 90656447 IC50 = 16870 nM T83875 C4P6YN 90656448 IC50 = 19230 nM T83875 CRM6W2 90656449 IC50 = 4310 nM T83875 C29OBX 90656450 IC50 = 1890 nM T83875 C3JTI2 90656451 IC50 = 11090 nM T83875 CNPR45 90656453 IC50 = 13780 nM T83875 CI8AN7 90656454 IC50 = 4580 nM T83875 C2DO3S 90656455 IC50 = 10930 nM T83875 CX2BI1 90665464 IC50 = 1560 nM T83875 C2U4IX 90665465 IC50 = 1810 nM T83875 CRB45O 90665466 IC50 = 2310 nM T83875 C3FLR5 90665467 IC50 = 1370 nM T83875 CQB95X 90665468 IC50 = 2450 nM T83875 CV53TJ 90665469 IC50 = 2930 nM T83875 C9S6WJ 90665470 IC50 = 15840 nM T83875 CX2J6R 90665471 IC50 = 2520 nM T83875 CY9HP0 90665472 IC50 = 2400 nM T83875 C1LYK6 90665473 IC50 = 6970 nM T83875 CVH28D 90665474 IC50 = 3690 nM T83875 C0BVY5 90665475 IC50 = 4130 nM T83875 CH8QE5 90665476 IC50 = 3910 nM T83875 C3VT2Z 90665477 IC50 = 1210 nM T83875 CDG71U 90665478 IC50 = 2600 nM T83875 COJ3I8 90665479 IC50 = 1910 nM T83875 CB2JY6 90665480 IC50 = 2010 nM T83875 CZ3K2I 90665481 IC50 = 1940 nM T83875 C98OBK 90665482 IC50 = 2330 nM T83875 CX1S7A 90665483 IC50 = 2910 nM T83875 CRLT57 90665484 IC50 = 2440 nM T83875 CR1IF2 90665485 IC50 = 2290 nM T83875 CUS3H7 90665486 IC50 = 3230 nM T83875 CZ2I3Q 90665487 IC50 = 3630 nM T83875 CXA4S3 90665488 IC50 = 2110 nM T83875 CQT26E 90665489 IC50 = 7070 nM T83875 C5LU6I 90665490 IC50 = 1770 nM T83875 CF4ZN3 90665491 IC50 = 2710 nM T83875 CAW89J 90665492 IC50 = 3730 nM T83875 C6NZ2T 90665493 IC50 = 6950 nM T83875 C4YHG6 90665494 IC50 = 2000 nM T83875 CCEG94 90665495 IC50 = 2570 nM T83875 CBE9W8 90665496 IC50 = 8670 nM T83875 CT81HP 90665497 IC50 = 5920 nM T83875 C1JCF4 90666201 IC50 = 16380 nM T83875 C0MNS2 90666203 IC50 = 6470 nM T83875 C53HVF 90666204 IC50 = 1680 nM T83875 C52ZRU 90666205 IC50 = 2670 nM T83875 CG7U0D 90666206 IC50 = 6520 nM T83875 CEM2C7 90666207 IC50 = 7650 nM T83875 CFD4H5 90666208 IC50 = 2390 nM T83875 C1YTP6 90666209 IC50 = 8290 nM T83875 C54YQR 90666210 IC50 = 8630 nM T83875 CHMD93 90666391 IC50 = 9180 nM T83875 CAS3P4 90667148 IC50 = 45970 nM T83875 CIX7G5 90676868 IC50 = 1070 nM T83875 C29MFT 90676892 IC50 = 271 nM T83875 CNC4Q0 91664024 IC50 > 10000 nM T83875 C1SZM3 91809224 IC50 = 60 nM T83875 C68YVN 91827407 IC50 > 200000 nM T83875 CZQ9E5 91863223 IC50 = 50700 nM T83875 C90AXQ 91863224 IC50 = 17700 nM T83875 C4GQ7A 91863375 IC50 > 100000 nM T83875 CL45WP 91863383 IC50 = 89050 nM T83875 C2XO9G 91973312 IC50 = 14 nM T83875 CK59LE 91973747 IC50 = 405 nM T83875 C58BTI 91973750 IC50 = 121 nM T83875 CU5D3W 93990915 IC50 = 9700 nM T83875 CF3I7E 96469773 IC50 = 1160 nM T83875 CMS13T 97182268 IC50 = 19600 nM T83875 C08XPB 101896439 IC50 = 2400 nM T83875 C85QZO 101896440 IC50 = 2000 nM T83875 C81WRJ 101910778 IC50 = 6.3 nM T83875 CQ1SM0 102004295 IC50 = 290 nM T83875 C7CR9D 102220645 IC50 = 10500 nM T83875 C3RW4H 102313434 IC50 > 100000 nM T83875 C0X7BR 107271816 IC50 > 10000 nM T83875 CR4W5N 110704124 IC50 > 10000 nM T83875 CB2JW9 114940252 IC50 = 7980 nM T83875 C8TX3R 115328020 IC50 = 1500 nM T83875 CQ8MX9 117929947 IC50 = 41373 nM T83875 CKWG83 117939777 IC50 = 125996 nM T83875 CL54XO 117939779 IC50 > 50000 nM T83875 C4D5QS 117939782 IC50 > 50000 nM T83875 CP07SU 117939783 IC50 > 50000 nM T83875 CM8A4Q 117939786 IC50 > 50000 nM T83875 CFYK36 117939787 IC50 > 50000 nM T83875 C3JB9W 117939792 IC50 > 50000 nM T83875 CW7PI3 117939793 IC50 > 50000 nM T83875 CE53IP 117939804 IC50 > 50000 nM T83875 C21BRF 117939805 IC50 > 50000 nM T83875 CMJF04 117939806 IC50 > 50000 nM T83875 C0HS3B 117939808 IC50 > 50000 nM T83875 CYW8F3 117939809 IC50 > 50000 nM T83875 C7QP6F 117939810 IC50 > 50000 nM T83875 C76QNR 117939811 IC50 > 50000 nM T83875 C75RLB 117939814 IC50 > 50000 nM T83875 C8W3YQ 117939815 IC50 > 50000 nM T83875 C4J5TP 117939817 IC50 = 217101 nM T83875 CL30GA 117939818 IC50 > 50000 nM T83875 CN6IS1 117939819 IC50 = 954993 nM T83875 CLU64K 117939825 IC50 > 50000 nM T83875 CW28FI 117939826 IC50 = 358922 nM T83875 CCS42Z 117945944 IC50 = 9500 nM T83875 CYBX18 118140875 IC50 = 3.7 nM T83875 C1J9DW 118140947 IC50 = 3.4 nM T83875 CN7I8Q 118297734 IC50 > 200000 nM T83875 C61BNV 118304877 IC50 > 10000 nM T83875 C2U3NT 118483746 IC50 = 70 nM T83875 C38WNG 118483913 IC50 = 94 nM T83875 C6A8FW 118483914 IC50 = 82.8 nM T83875 CF7Z1S 118493308 IC50 > 10000 nM T83875 C10VNP 118536083 IC50 = 54.8 nM T83875 CF90SQ 118536088 IC50 = 193.1 nM T83875 C9T8ZB 118536101 IC50 = 687.1 nM T83875 C72EDN 118536105 IC50 = 589.6 nM T83875 CYHM83 118536120 IC50 = 29.7 nM T83875 C9BUT8 118536122 IC50 = 90.5 nM T83875 CY2JZ4 118542609 IC50 = 160 nM T83875 CC95BW 118706231 Ki = 45 nM T83875 CT1O7D 118706232 Ki = 91 nM T83875 CMS52X 118706233 Ki = 34 nM T83875 C3UE9R 118706234 Ki = 12 nM T83875 CUFL29 118706235 Ki = 10 nM T83875 C3M4SH 118706236 Ki = 12 nM T83875 CY5DO8 118706237 Ki = 34 nM T83875 C4VA3Z 118706239 Ki = 41 nM T83875 C3AY6U 118709465 IC50 > 10000 nM T83875 C87JAX 118709466 IC50 > 10000 nM T83875 CCH7X5 118709467 IC50 > 10000 nM T83875 C1BF7M 118709468 IC50 > 10000 nM T83875 CU2Y0H 118709469 IC50 > 10000 nM T83875 C4H1TQ 118712953 IC50 = 527 nM T83875 C4J8TS 118712954 IC50 = 1300 nM T83875 CH0YP2 118712955 IC50 = 21.4 nM T83875 C2BZ4I 118712956 IC50 = 1280 nM T83875 CR34TU 118718853 IC50 = 15510 nM T83875 CX93MC 118724438 IC50 = 4180 nM T83875 C57BEW 118726138 IC50 = 6000 nM T83875 CUVW23 118726139 IC50 = 5220 nM T83875 C2UX0J 118726140 IC50 = 12710 nM T83875 C1WGY9 118726141 IC50 = 11320 nM T83875 C7GXD9 118726142 IC50 = 9510 nM T83875 CZ28ED 118726143 IC50 = 8020 nM T83875 C3A2XO 118726144 IC50 = 7250 nM T83875 CQ5N0W 118726145 IC50 = 9650 nM T83875 C1IBC8 118726146 IC50 = 14400 nM T83875 CYPE42 118726147 IC50 = 3720 nM T83875 CDX5V0 118726148 IC50 = 6010 nM T83875 C0EXZ7 118726149 IC50 = 24520 nM T83875 C2GPM3 118726150 IC50 = 20010 nM T83875 CUZ38P 118726151 IC50 = 23160 nM T83875 CNY9K4 118726152 IC50 = 16860 nM T83875 CC87QU 118726153 IC50 = 21200 nM T83875 CTBQ68 118726154 IC50 = 18330 nM T83875 CY5H2Q 118726155 IC50 = 27010 nM T83875 CZ8DR0 118726156 IC50 = 24300 nM T83875 C8PRQ1 118726157 IC50 = 31240 nM T83875 C1TR3D 118726161 IC50 = 26280 nM T83875 C3COH5 118726165 IC50 = 10470 nM T83875 CN4GY5 118726166 IC50 = 13080 nM T83875 CUT7H1 118726167 IC50 = 30300 nM T83875 CIZ8P9 118726168 IC50 = 7800 nM T83875 CO3N6F 118726169 IC50 = 8380 nM T83875 CSJR39 118726170 IC50 = 12290 nM T83875 C2PC1W 118726171 IC50 = 12440 nM T83875 C17VOQ 118726172 IC50 = 25650 nM T83875 C4VX5E 118727528 IC50 = 129 nM T83875 C1LK6U 118727529 IC50 = 19400 nM T83875 C6PX9T 118727530 IC50 = 35 nM T83875 C3HD8M 118727531 IC50 = 3480 nM T83875 CADH94 118727532 IC50 = 726 nM T83875 C9G1YD 118727533 IC50 = 2190 nM T83875 CRN59D 118727534 IC50 > 100000 nM T83875 CTH6S4 118727535 IC50 = 4 nM T83875 CY8Q9V 118727536 IC50 = 118 nM T83875 CP7A9D 118727537 IC50 = 142 nM T83875 CFWJ56 118728390 IC50 > 100000 nM T83875 CMEA81 118728391 IC50 > 100000 nM T83875 CJ8ZY2 118728392 IC50 > 100000 nM T83875 CW8Z2H 118728853 IC50 > 100000 nM T83875 C9XEY8 118728854 IC50 > 100000 nM T83875 CVCT10 118728855 IC50 > 100000 nM T83875 C1JX3S 118728856 IC50 > 100000 nM T83875 CULF09 118728857 IC50 > 100000 nM T83875 CDKA92 118728858 IC50 > 100000 nM T83875 C4XUG3 118728859 IC50 > 100000 nM T83875 CK3E9J 118728860 IC50 > 100000 nM T83875 C8L6TZ 118728861 IC50 > 100000 nM T83875 CS8UI6 118728862 IC50 > 100000 nM T83875 CAZ78X 118728978 IC50 = 87700 nM T83875 CXG4B7 118728979 IC50 = 77100 nM T83875 C7UED4 118728980 IC50 = 36000 nM T83875 CK9AX4 118728981 IC50 = 13200 nM T83875 C68EHZ 118728982 IC50 = 16900 nM T83875 C1LY8F 118728983 IC50 = 27800 nM T83875 CVP9F5 118728984 IC50 = 70400 nM T83875 CXOA52 118730192 IC50 = 257.6 nM T83875 C27ZWI 118730193 IC50 = 9100 nM T83875 CEQ56Z 118730194 IC50 = 19200 nM T83875 C3D6VY 118730195 IC50 = 45300 nM T83875 CJ2P9D 118730196 IC50 = 876.6 nM T83875 CI2X8N 118730197 IC50 = 9100 nM T83875 CP70TH 118730198 IC50 = 10300 nM T83875 CPAT89 118730199 IC50 = 630100 nM T83875 C5F4LP 118730200 IC50 = 310600 nM T83875 CD21PC 118731187 IC50 = 1300 nM T83875 C07UCB 118733540 IC50 = 0.85 nM T83875 CM76SB 118733551 IC50 = 370 nM T83875 C6RY3J 118734094 IC50 = 39 nM T83875 CY57TV 118734096 IC50 = 1370 nM T83875 C0SR8X 118734098 IC50 = 1540 nM T83875 C0J2WE 118734102 IC50 = 37 nM T83875 CW81OF 118734104 IC50 = 25 nM T83875 CCN86A 118734106 IC50 = 650 nM T83875 CH7OT9 118734108 IC50 = 70 nM T83875 C3XB0N 118734706 IC50 = 21950 nM T83875 C67ZXU 118734710 IC50 = 78590 nM T83875 CNB83Q 118734712 IC50 = 53070 nM T83875 CX80VO 118734713 IC50 = 15070 nM T83875 CDO43K 118734715 IC50 = 66740 nM T83875 C67CLN 118734716 IC50 = 6050 nM T83875 C5SN4X 118734717 IC50 = 10350 nM T83875 CSDJ67 118734721 IC50 = 6020 nM T83875 CN3S6M 118734722 IC50 = 9180 nM T83875 C7Y0LX 118735096 IC50 = 110 nM T83875 C8QOE4 118735098 IC50 = 200 nM T83875 C41EPX 118913669 IC50 > 100000 nM T83875 CJ5NC9 118913682 IC50 > 100000 nM T83875 C1ENW9 118913743 IC50 = 24900 nM T83875 CQNM60 118918087 IC50 = 47200 nM T83875 CGZ1L3 118931167 IC50 = 41300 nM T83875 CMX4J6 121482363 IC50 > 50000 nM T83875 CD9H0B 122179917 IC50 = 3410 nM T83875 C9P1NG 122179918 IC50 = 5530 nM T83875 CK3T9I 122179919 IC50 = 5370 nM T83875 C3ZST9 122179922 IC50 = 1020 nM T83875 C6EZH1 122179924 IC50 = 700 nM T83875 C6C5YK 122179927 IC50 = 1030 nM T83875 C6PTD5 122180404 IC50 = 480 nM T83875 C1X9KB 122180406 IC50 = 390 nM T83875 CMC26Y 122180416 IC50 = 191 nM T83875 C8UIY9 122180417 IC50 = 115 nM T83875 CJK24Z 122180436 IC50 = 4300 nM T83875 CKM1E7 122180462 IC50 = 15800 nM T83875 CMD2B6 122180465 IC50 = 13000 nM T83875 C79SBR 122180468 IC50 = 4480 nM T83875 CM2PD5 122186418 IC50 = 67300 nM T83875 C1V5AO 122186419 IC50 = 1500 nM T83875 CQ5PO2 122186420 IC50 = 4900 nM T83875 CD0V5N 122186421 IC50 = 5100 nM T83875 C4L3WE 122186422 IC50 = 1600 nM T83875 C21HOI 122186423 IC50 = 1700 nM T83875 CH35KZ 122186425 IC50 = 120 nM T83875 C03TJD 122186427 IC50 = 250 nM T83875 CEVY24 122186429 IC50 = 220 nM T83875 CC91RU 122186431 IC50 = 3200 nM T83875 CO0B7A 122186433 IC50 = 7300 nM T83875 CM94AW 122186435 IC50 = 14600 nM T83875 CA4M3I 122186437 IC50 = 22500 nM T83875 C8YIT5 122186439 IC50 = 4500 nM T83875 C2PC4U 122186440 IC50 = 1200 nM T83875 CZS2M9 122186441 IC50 = 510 nM T83875 C5VNO0 122186442 IC50 = 3500 nM T83875 CZ5B7W 122186443 IC50 = 6300 nM T83875 CA4GO3 122188866 IC50 > 100000 nM T83875 CNYA71 122188867 IC50 = 9220 nM T83875 CCEQ57 122188868 IC50 > 100000 nM T83875 CHK2M9 122188869 IC50 > 100000 nM T83875 C5SNF1 122188870 IC50 > 100000 nM T83875 C1K0PT 122188871 IC50 > 100000 nM T83875 COM53A 122194326 IC50 = 41700 nM T83875 C2E6HQ 122194327 IC50 > 60000 nM T83875 C05DBN 122194328 IC50 > 60000 nM T83875 CYHF09 122194329 IC50 > 60000 nM T83875 C16GMN 122194330 IC50 > 60000 nM T83875 CS1UH0 122194331 IC50 > 60000 nM T83875 CN9CU1 122194332 IC50 = 58190 nM T83875 CTED74 122194333 IC50 = 30390 nM T83875 C8ZPO0 122194334 IC50 = 44270 nM T83875 C0B7ED 122194335 IC50 > 60000 nM T83875 CI9F4S 122194603 IC50 > 60000 nM T83875 C4MQP9 122194604 IC50 > 60000 nM T83875 CU1HE5 122194605 IC50 = 3010 nM T83875 CV5RC2 122194606 IC50 = 12110 nM T83875 C4OEV3 122194607 IC50 = 3200 nM T83875 CR62NI 122194608 IC50 = 7070 nM T83875 C8VQA9 122194609 IC50 = 21200 nM T83875 CHRQ34 122194610 IC50 > 60000 nM T83875 CSZ72C 122194611 IC50 = 5300 nM T83875 CLZ8S5 122194612 IC50 = 60000 nM T83875 CA79DS 122415289 IC50 > 50000 nM T83875 CM7R6T 123440770 IC50 = 50200 nM T83875 C9U0EL 124115926 IC50 = 1200 nM T83875 C5WHS1 124116114 IC50 = 1670 nM T83875 CR81DC 124116115 IC50 = 741 nM T83875 C01TOU 124116118 IC50 = 157 nM T83875 C8U5RC 124313549 IC50 > 100000 nM T83875 CI5M3O 126842840 IC50 = 16000 nM T83875 C6N1OH 127025105 IC50 = 2195 nM T83875 C3YK6S 127025108 IC50 = 53260 nM T83875 C21OBG 127025662 IC50 = 4712 nM T83875 C9H5EW 127025664 IC50 = 4756 nM T83875 CL3RP0 127025669 IC50 = 4055 nM T83875 C6GNR7 127026321 IC50 = 55680 nM T83875 CN0A5U 127026324 IC50 = 3904 nM T83875 CNR05U 127027039 Ki > 50000 nM T83875 C8WJF6 127027348 Ki > 50000 nM T83875 CT6AD7 127027787 IC50 = 4654 nM T83875 C5A9ZJ 127028005 Ki > 50000 nM T83875 C5IGO0 127028297 Ki > 50000 nM T83875 C19THR 127030340 IC50 = 115 nM T83875 CDL0C7 127031303 IC50 > 100000 nM T83875 CLT4M1 127031655 IC50 = 40 nM T83875 CJ2U6F 127032119 IC50 = 457 nM T83875 C0C9WI 127032253 IC50 = 25 nM T83875 CQT5M1 127034333 IC50 = 344.7 nM T83875 COY03I 127034334 IC50 = 999.8 nM T83875 C69KJB 127034561 IC50 = 27.9 nM T83875 C9RB7W 127035092 IC50 = 8090 nM T83875 C94YFD 127035093 IC50 = 6670 nM T83875 CGDB19 127035094 IC50 = 43930 nM T83875 C3LJ9W 127035097 IC50 = 20750 nM T83875 CG5SI3 127035266 IC50 = 15300 nM T83875 CC45DE 127035495 IC50 = 260 nM T83875 C9SEO1 127035497 IC50 = 110 nM T83875 CN1JC8 127035507 IC50 = 160 nM T83875 C2DL5A 127035509 IC50 = 460 nM T83875 C9GMF4 127035552 IC50 = 34890 nM T83875 CMP1D6 127035554 IC50 = 15770 nM T83875 CG70KY 127035960 IC50 = 3810 nM T83875 C1XAW5 127035961 IC50 = 267000 nM T83875 CB5W1U 127035962 IC50 = 9990 nM T83875 CS4B8G 127036275 IC50 = 19460 nM T83875 C5SUJ2 127036479 IC50 = 26730 nM T83875 CUZR67 127036672 IC50 = 16100 nM T83875 CWDI07 127037076 IC50 = 143000 nM T83875 CL29WO 127037458 IC50 = 8980 nM T83875 C0S8GJ 127037470 IC50 = 40580 nM T83875 C2W4DY 127037999 IC50 = 144200 nM T83875 CN3QG5 127038898 IC50 = 21300 nM T83875 C3C4UD 127042054 IC50 = 46550 nM T83875 C9US1F 127042057 IC50 = 115200 nM T83875 C1NB5G 127042331 IC50 > 100000 nM T83875 CF7BE1 127042742 IC50 = 111660 nM T83875 CN6HZ3 127042941 IC50 = 189 nM T83875 C3Z8FA 127042942 IC50 = 2550 nM T83875 CJ6W2U 127045743 IC50 = 6920 nM T83875 CGUC67 127045964 IC50 = 522 nM T83875 C4DRT5 127046073 IC50 > 100000 nM T83875 CT0DZ1 127046074 IC50 > 100000 nM T83875 CXP8S3 127046075 IC50 > 100000 nM T83875 C71PDE 127046206 IC50 > 100000 nM T83875 C5KOC8 127046207 IC50 > 100000 nM T83875 C4MOG6 127046208 IC50 > 100000 nM T83875 CTDZ75 127046395 IC50 = 19000 nM T83875 CTVO57 127046396 IC50 = 1750 nM T83875 CG8X9O 127046431 IC50 = 6350 nM T83875 CW51KH 127046559 IC50 = 147 nM T83875 C5P7UB 127046560 IC50 = 1130 nM T83875 CI7AO8 127046561 IC50 > 100000 nM T83875 CYNG69 127046593 IC50 > 100000 nM T83875 CH4MZ0 127046738 IC50 > 100000 nM T83875 CIK0O4 127046739 IC50 = 2080 nM T83875 C3H2TR 127046740 IC50 = 23300 nM T83875 C75RDT 127046765 IC50 = 2110 nM T83875 CC14IO 127047102 IC50 = 1240 nM T83875 CHQ3V7 127047235 IC50 = 250 nM T83875 CC4R1Z 127047236 IC50 = 5380 nM T83875 C90YDX 127047237 IC50 = 661 nM T83875 CREG96 127047238 IC50 = 6120 nM T83875 CU39GI 127047239 IC50 = 5510 nM T83875 CN46VR 127047342 IC50 > 100000 nM T83875 CCS71F 127047626 IC50 = 4990 nM T83875 CW7A9C 127047746 IC50 = 6700 nM T83875 CZ1L4H 127047856 IC50 = 5120 nM T83875 C9EML8 127047875 IC50 > 100000 nM T83875 CW2B3M 127048716 IC50 = 57500 nM T83875 C23EOB 127049071 IC50 = 3500 nM T83875 CU85GC 127049730 IC50 = 11400 nM T83875 C83LIY 129165316 IC50 > 10000 nM T83875 CJGE94 129165458 IC50 > 10000 nM T83875 C84UJE 130302628 IC50 > 30000 nM T83875 C3M2IV 130344977 IC50 = 88300 nM T83875 CE8Q7I 130345035 IC50 > 100000 nM T83875 C01UGK 130345060 IC50 = 29200 nM T83875 CN9S7B 130345097 IC50 > 100000 nM T83875 C3CH7B 130345110 IC50 > 100000 nM T83875 C7RN8L 130345158 IC50 = 33000 nM T83875 CF20BS 130345178 IC50 = 59300 nM T83875 CMO50A 130345200 IC50 > 100000 nM T83875 C29WVS 130358344 IC50 > 100000 nM T83875 CZM13E 130358354 IC50 = 61700 nM T83875 CW47IH 130638185 IC50 = 4100 nM T83875 CP8L7V 132137973 IC50 = 45840 nM T83875 CRG1Y4 132342060 IC50 > 100000 nM T83875 CZ3OD0 132495360 IC50 > 100000 nM T83875 CBN5C0 132495361 IC50 > 100000 nM T83875 C2CJF3 132503347 IC50 = 5120 nM T83875 C7DC2X 132511215 IC50 = 32000 nM T83875 C0ERW7 132511218 IC50 > 100000 nM T83875 CL9UY5 132511220 IC50 > 100000 nM T83875 CL23KG 132571526 IC50 = 440 nM T83875 CF3X5S 132577022 IC50 > 500000 nM T83875 C1TJ7B 132578491 IC50 > 10000 nM T83875 C5CKG0 132578492 IC50 > 10000 nM T83875 CYB73H 132579936 IC50 > 500000 nM T83875 CF3M0N 132579937 IC50 = 97100 nM T83875 C9MRW2 132579938 IC50 = 500 nM T83875 CGIQ08 132579939 IC50 = 27400 nM T83875 C87SOL 132961376 IC50 = 1010 nM T83875 C6U1LV 132969040 Ki = 5700 nM T83875 C45WQG 132969041 Ki = 6000 nM T83875 CL6XW8 132969042 Ki = 2180 nM T83875 CF4OX9 134131513 IC50 = 10200 nM T83875 CBJ3G2 134131700 IC50 = 3610 nM T83875 CCJF74 134132255 IC50 = 1600 nM T83875 CG1TY4 134132538 IC50 = 961 nM T83875 CRY9P0 134133186 IC50 = 2080 nM T83875 CHT37D 134133216 IC50 = 1940 nM T83875 C6VS5U 134133379 IC50 > 100000 nM T83875 CVF3T5 134133384 IC50 = 10200 nM T83875 CSA09I 134137557 IC50 = 35600 nM T83875 C97CUD 134137716 IC50 = 46500 nM T83875 CV3J2Q 134138913 IC50 = 679 nM T83875 CF76XM 134139033 IC50 = 1330 nM T83875 CQU8T5 134139124 IC50 > 100000 nM T83875 CJ6AO0 134139236 IC50 > 100000 nM T83875 C51HUD 134140107 Ki = 2480 nM T83875 CF9C1X 134140379 IC50 = 1190 nM T83875 C73LGF 134140781 IC50 > 100000 nM T83875 CFJ74X 134140944 IC50 = 235 nM T83875 CSYM31 134142478 IC50 > 100000 nM T83875 CUP09Q 134142596 IC50 > 100000 nM T83875 C0S6OI 134142875 Ki = 2810 nM T83875 C47KWL 134144584 IC50 > 100000 nM T83875 CP0D4F 134146126 IC50 > 100000 nM T83875 CZM9O4 134146757 IC50 = 4500 nM T83875 C3RHY4 134147228 IC50 = 1050 nM T83875 C7E3YA 134149382 IC50 > 100000 nM T83875 C0V3GR 134149702 IC50 = 9240 nM T83875 CJ1D3P 134149885 IC50 = 458 nM T83875 C4Y5ZX 134150471 IC50 = 5500 nM T83875 CRZ2W4 134150858 IC50 > 100000 nM T83875 C8XJH0 134151923 IC50 = 131 nM T83875 CJ98WY 134152913 IC50 > 100000 nM T83875 CF8RV4 134153109 IC50 = 444 nM T83875 CA2KR0 134153338 IC50 = 12200 nM T83875 CPBG73 134153558 IC50 > 100000 nM T83875 C95UFC 134154267 IC50 = 29700 nM T83875 CGK4X3 134155114 IC50 = 860 nM T83875 C9QXG2 134155279 IC50 = 37000 nM T83875 CQA14Y 134155772 IC50 > 100000 nM T83875 C07ZGI 134156270 IC50 = 3220 nM T83875 C9A2GK 134156912 Ki = 1140 nM T83875 CC0IG7 134157232 IC50 > 100000 nM T83875 CK1C8S 134366896 IC50 = 19927.3 nM T83875 C67XBZ 134366929 IC50 = 5927.3 nM T83875 C5TES6 134366930 IC50 = 75779.6 nM T83875 CD0B8J 134366950 IC50 = 129064 nM T83875 CCX21V 134366961 IC50 = 162399.3 nM T83875 C59ORQ 134366996 IC50 = 21478.3 nM T83875 C83FUK 134385636 IC50 = 6906.8 nM T83875 C0CU9Q 134385638 IC50 = 66028.4 nM T83875 CFU6H7 134385639 IC50 > 100000 nM T83875 CP8VX4 134385640 IC50 = 32960.7 nM T83875 C6HB5G 134385645 IC50 = 27293.2 nM T83875 C9QZH6 134385648 IC50 = 73638.2 nM T83875 CK6L7Y 134385649 IC50 = 20564.5 nM T83875 C9LNR7 134816193 IC50 = 370 nM T83875 CA2H1G 134816270 IC50 > 10000 nM T83875 CEYR15 134816271 IC50 > 10000 nM T83875 CTOB53 134816331 IC50 > 10000 nM T83875 C2X3GF 134816595 IC50 > 10000 nM T83875 CD9B4Z 134816640 IC50 > 10000 nM T83875 C35ZVJ 134816641 IC50 = 50 nM T83875 C4R6KL 134816691 IC50 > 10000 nM T83875 C0IOP2 134816692 IC50 > 10000 nM T83875 CC94YQ 134816693 IC50 > 10000 nM T83875 CP86GA 134816695 IC50 > 10000 nM T83875 CUD08L 134817200 IC50 = 145 nM T83875 C2ATF7 135401432 IC50 = 2783 nM T83875 C0UCX3 135408731 IC50 > 10000 nM T83875 C5T9YE 135436602 IC50 = 10 nM T83875 C8WL0I 135449090 IC50 = 98 nM T83875 C2WA9R 135457295 Ki = 2 nM T83875 CGFS08 135459067 IC50 > 100000 nM T83875 CTE23K 135464118 IC50 = 5867 nM T83875 CB53EI 135465870 IC50 = 3075 nM T83875 CHNA50 135471217 IC50 = 10 nM T83875 C7AGR0 135474338 IC50 = 165 nM T83875 CJR38B 135483618 IC50 = 8 nM T83875 CKG25Y 135495099 IC50 = 9 nM T83875 CT3M5A 135497038 IC50 = 10 nM T83875 CCDS87 135499808 IC50 = 8.6 nM T83875 C34FXW 135501716 IC50 = 1233 nM T83875 C71EOH 135511237 Ki = 130000 nM T83875 C6VS7P 135514579 IC50 = 100 nM T83875 C1CZ9M 135514796 IC50 = 12750 nM T83875 CR05TL 135516788 Ki = 4 nM T83875 CD2X0Y 135524872 IC50 = 9 nM T83875 C5UO1D 135679868 Ki = 130000 nM T83875 CY57UW 135719318 IC50 = 3120 nM T83875 C60MRN 135719324 IC50 = 2340 nM T83875 CCNH91 135743577 IC50 > 300000 nM T83875 CZ97SK 135778696 IC50 = 88500 nM T83875 C03HVY 135846955 IC50 = 1967 nM T83875 CQCT18 135846958 IC50 = 6075 nM T83875 CE4QG5 135846981 IC50 = 5817 nM T83875 C3UB7L 135846982 IC50 = 1123 nM T83875 CKDW41 135966009 IC50 = 14333 nM T83875 CPH2S1 136059661 IC50 = 5560 nM T83875 COE97S 136066029 IC50 = 32100 nM T83875 C2L8UX 136074346 Ki = 130 nM T83875 C8E2KH 136074347 Ki = 10 nM T83875 CX95EP 136092233 IC50 = 9 nM T83875 CA3JC8 136118613 IC50 = 1517 nM T83875 CQ2GP6 136118614 IC50 = 327 nM T83875 C6R4IC 136118615 IC50 = 1197 nM T83875 CS0JL5 136118616 IC50 = 2583 nM T83875 C8RH6M 136118617 IC50 = 263 nM T83875 CN4U6K 136118618 IC50 = 29 nM T83875 CHWC38 136118619 IC50 = 1900 nM T83875 C5UDW3 136118620 IC50 = 2067 nM T83875 C8I6UN 136118621 IC50 = 52 nM T83875 CV4E6W 136118635 IC50 = 267 nM T83875 CFI2X7 136118636 IC50 = 1533 nM T83875 CYS3M8 136118637 IC50 = 543 nM T83875 C0UH1B 136118638 IC50 = 677 nM T83875 C6G4AY 136118639 IC50 = 7133 nM T83875 C40VES 136118640 IC50 = 533 nM T83875 CH4Q8O 136118646 IC50 = 627 nM T83875 C43JTG 136118647 IC50 = 13333 nM T83875 CLH0V9 136118648 IC50 = 1800 nM T83875 C76XEJ 136118649 IC50 = 1200 nM T83875 CN0V5C 136118650 IC50 = 4433 nM T83875 CR72MQ 136118651 IC50 = 3900 nM T83875 CD7OE2 136118652 IC50 = 5475 nM T83875 CG5TX8 136118653 IC50 = 3250 nM T83875 CCHM67 136118657 IC50 = 1080 nM T83875 C0W1TM 136118658 IC50 = 623 nM T83875 C40LYH 136118659 IC50 = 85 nM T83875 CZ7C3Y 136118660 IC50 = 18 nM T83875 C42FCS 136118661 IC50 = 153 nM T83875 CR3DK1 136118716 IC50 = 2467 nM T83875 CON04G 136118728 IC50 = 3683 nM T83875 COX1F8 136118729 IC50 = 5517 nM T83875 CY5GU4 136118730 IC50 = 26167 nM T83875 C0R5PV 136118732 IC50 = 6107 nM T83875 CLU47S 136203753 IC50 = 316.23 nM T83875 CUD85K 136215758 Ki = 150000 nM T83875 C5SH0A 136219375 Ki = 880 nM T83875 C4RP7K 136219376 Ki = 250 nM T83875 C3AIC2 136233006 IC50 = 16330 nM T83875 C7MLI3 136233007 IC50 = 9130 nM T83875 CK68XF 136233008 IC50 = 11820 nM T83875 CS81JR 136233009 IC50 = 18690 nM T83875 CE76VG 136233010 IC50 = 12730 nM T83875 C8KWN7 136233016 IC50 = 21870 nM T83875 CNGU52 136233017 IC50 = 810 nM T83875 CQK12T 136233018 IC50 = 3980 nM T83875 C9LR0M 136233021 IC50 = 1100 nM T83875 C20ULD 136233022 IC50 = 420 nM T83875 CI1XO6 136233023 IC50 = 1390 nM T83875 CPZ80S 136239406 Ki = 310 nM T83875 CEPX06 136239508 Ki = 810 nM T83875 CAB79P 136241665 IC50 > 200000 nM T83875 C5W8GX 136242978 Ki = 30 nM T83875 CT7LY9 136242979 Ki = 4 nM T83875 C6K3SZ 136244520 Ki = 760 nM T83875 C8XZR1 136260489 Ki = 610 nM T83875 CXM62D 136270607 Ki = 3870 nM T83875 CFP60G 136607463 IC50 = 132000 nM T83875 CHP3N6 136986940 Ki = 600 nM T83875 C0ORN6 136986942 Ki = 110 nM T83875 C0GT6R 136986944 Ki = 12 nM T83875 CD1EU8 136986946 Ki = 4670 nM T83875 CX4CS1 136986948 Ki = 240 nM T83875 C5GHZ1 136986950 Ki = 180 nM T83875 CU2T7W 136986952 Ki = 450 nM T83875 CVA2W6 136986954 Ki = 40 nM T83875 C1HI9Q 136986956 Ki = 79220 nM T83875 C6TYF4 137174990 Ki = 5020 nM T83875 C4ZKC3 137175204 Ki = 4250 nM T83875 C5A8RL 137175205 Ki = 550 nM T83875 C1PE4I 137175206 Ki = 60 nM T83875 CKS92O 137175207 Ki = 290 nM T83875 C36LNB 137175235 Ki = 440 nM T83875 C2FMA0 137175236 Ki = 2160 nM T83875 C7YZF2 137175237 Ki = 2580 nM T83875 CVP1K0 137175238 Ki = 9550 nM T83875 C9P4YE 137459864 IC50 > 31622.78 nM T83875 CIP6T2 137631403 IC50 = 6630 nM T83875 CLVQ93 137631579 IC50 > 10000 nM T83875 CE6L8G 137631680 IC50 = 53513 nM T83875 C74HIO 137631707 IC50 = 3090 nM T83875 CW0BZ8 137631800 IC50 = 9360 nM T83875 C9BXC6 137632300 IC50 = 620 nM T83875 CELH07 137632760 IC50 = 6460 nM T83875 C7TB1N 137633079 IC50 = 9586 nM T83875 CP43GR 137633264 IC50 = 9000 nM T83875 CZ2HK3 137633315 IC50 > 100000 nM T83875 CDA65L 137633416 IC50 > 100000 nM T83875 C1D9FT 137633537 IC50 = 8200 nM T83875 CPEG26 137633844 IC50 = 720 nM T83875 C6XUF8 137633971 IC50 = 1250 nM T83875 C7WEV4 137634210 IC50 = 14300 nM T83875 C0C6NP 137634473 IC50 >= 1000000 nM T83875 CM2CR5 137635058 IC50 = 7240 nM T83875 C8IZ6F 137635535 IC50 = 6310 nM T83875 C20CWR 137635957 IC50 = 6260 nM T83875 CBQ27R 137636063 IC50 = 8170 nM T83875 CF6ZK2 137636117 IC50 = 1130 nM T83875 C4LS1I 137636518 IC50 = 1030 nM T83875 C31QAB 137636695 IC50 = 5700 nM T83875 CB08HD 137636701 IC50 = 1940 nM T83875 CU4A5C 137636900 IC50 >= 1000000 nM T83875 COZ4G1 137636952 IC50 = 6800 nM T83875 CU5T9E 137636999 IC50 > 100000 nM T83875 CM35CX 137637171 IC50 > 100000 nM T83875 C9KOA0 137637296 IC50 > 100000 nM T83875 C0N3UQ 137637571 IC50 = 20800 nM T83875 CNEH91 137637802 IC50 = 8400 nM T83875 CIH2B0 137637832 IC50 > 100000 nM T83875 CBZ3T5 137638261 IC50 = 6600 nM T83875 CC85LZ 137638918 IC50 > 100000 nM T83875 CQ8IR3 137638955 IC50 > 100000 nM T83875 C9CYA8 137639104 IC50 > 100000 nM T83875 CY6VP5 137639127 IC50 > 25000 nM T83875 C70NHU 137639458 IC50 = 570 nM T83875 C3XP6B 137639555 IC50 >= 100000 nM T83875 C20ZJX 137640020 IC50 = 5600 nM T83875 C29UYV 137640667 IC50 = 2150 nM T83875 CVF68A 137640689 IC50 = 6780 nM T83875 C5ZV1Y 137640778 IC50 = 2790 nM T83875 CV20WQ 137641088 IC50 = 9300 nM T83875 C0CDW6 137641345 IC50 = 2400 nM T83875 CRS6D9 137641513 IC50 = 5940 nM T83875 C8GYQ2 137642138 IC50 > 100000 nM T83875 COX50U 137642409 IC50 = 1440 nM T83875 C7P6FH 137642777 IC50 >= 100000 nM T83875 COW6Y8 137643059 IC50 > 100000 nM T83875 C68RZL 137643060 IC50 > 100000 nM T83875 CL7K3X 137643291 IC50 > 10000 nM T83875 CR4PY5 137643351 IC50 = 1420 nM T83875 C1E9CL 137644000 IC50 = 7700 nM T83875 C4AGP8 137644230 IC50 = 3830 nM T83875 CC03ZF 137644660 IC50 > 100000 nM T83875 C0O2BL 137644693 IC50 > 100000 nM T83875 CAC64D 137645994 IC50 = 15650 nM T83875 CUG5D3 137646552 IC50 = 8570 nM T83875 C0P8ED 137646555 IC50 = 8900 nM T83875 CR60SF 137646770 IC50 = 1200 nM T83875 CMX01E 137646776 IC50 = 9400 nM T83875 CG1P3T 137646871 IC50 > 100000 nM T83875 C0OEH1 137647178 IC50 = 4650 nM T83875 C97WYL 137647179 IC50 > 100000 nM T83875 C4A6GE 137647180 IC50 > 100000 nM T83875 CTA0J8 137647190 IC50 = 600 nM T83875 C1D8NJ 137647314 IC50 >= 100000 nM T83875 C5RLG0 137647656 IC50 = 27075 nM T83875 C4VQK8 137648638 IC50 = 1540 nM T83875 CSO5A1 137648685 IC50 = 9810 nM T83875 C3WG5E 137649658 IC50 = 19606 nM T83875 CO3E6R 137649886 IC50 = 7400 nM T83875 C03HQU 137649999 IC50 = 3180 nM T83875 CG4XY5 137650246 IC50 = 2720 nM T83875 CR61GZ 137650279 IC50 = 1300 nM T83875 C0S8OQ 137650303 IC50 = 11800 nM T83875 CZ96CG 137650801 IC50 = 11400 nM T83875 CSD27L 137651785 IC50 > 100000 nM T83875 C5LMU7 137651876 IC50 = 7140 nM T83875 C4UG6F 137651890 IC50 > 100000 nM T83875 CFXL04 137652113 IC50 = 2819 nM T83875 CQ9B8K 137652578 IC50 = 570 nM T83875 CQ84TK 137652979 IC50 > 100000 nM T83875 C4AET5 137653036 IC50 >= 100000 nM T83875 C7ANF0 137653292 IC50 = 1300 nM T83875 C6R2QD 137653751 IC50 = 1000 nM T83875 C9NKO3 137653809 IC50 = 8780 nM T83875 CES62O 137653949 IC50 = 43317 nM T83875 CS46QP 137654687 IC50 = 7350 nM T83875 CG0YV5 137655066 IC50 = 9600 nM T83875 C38WAR 137655553 IC50 = 13200 nM T83875 CA1K3D 137655576 IC50 = 5400 nM T83875 C6RN4D 137655667 IC50 = 4200 nM T83875 C9Q4BS 137655777 IC50 > 100000 nM T83875 C0R6HE 137655915 IC50 = 340 nM T83875 CTM8B1 137656100 IC50 > 10000 nM T83875 CUZJ29 137656171 IC50 = 7270 nM T83875 CK93UH 137656494 IC50 = 4400 nM T83875 C4F2WI 137656817 IC50 > 100000 nM T83875 CJL6G1 137657126 IC50 = 1650 nM T83875 C79ECM 137657666 IC50 = 4550 nM T83875 C81NJW 137657973 IC50 = 8400 nM T83875 C0VPL8 137658080 IC50 > 100000 nM T83875 CB6DH1 137658226 IC50 = 6340 nM T83875 CQ1G8S 137658745 IC50 = 6900 nM T83875 CUT45L 137658804 IC50 = 6200 nM T83875 CZP1H6 137658871 IC50 = 15200 nM T83875 C6XDF0 137658917 IC50 >= 1000000 nM T83875 C0X6QO 137659176 IC50 = 9400 nM T83875 CFD5A3 137659177 IC50 >= 1000000 nM T83875 CZL1Y8 137659445 IC50 > 100000 nM T83875 C7UHX3 137659615 IC50 = 1020 nM T83875 C4NAO0 137659819 IC50 = 3350 nM T83875 CG3M6F 137660472 IC50 = 2620 nM T83875 CE0VO7 137660963 IC50 = 3340 nM T83875 CS2W1X 137661035 IC50 = 16000 nM T83875 CSM2V9 137661192 IC50 = 19320 nM T83875 C9VSC4 137661292 IC50 = 4470 nM T83875 C57MXQ 137661372 IC50 > 100000 nM T83875 CSU21O 137661504 IC50 = 1000 nM T83875 CJS6U1 137662125 IC50 > 100000 nM T83875 C16IHB 137662240 IC50 = 851 nM T83875 CQ5W3D 139449915 IC50 > 100000 nM T83875 CMG0D5 141488053 IC50 = 14090 nM T83875 CIN08E 141520106 IC50 = 7630 nM T83875 CR8W6O 141520108 IC50 > 200000 nM T83875 CN1TV3 141520110 IC50 = 98490 nM T83875 CFYM37 141520115 IC50 = 2460 nM T83875 C0R3XT 141520119 IC50 = 89950 nM T83875 C02TUS 141520121 IC50 = 110700 nM T83875 CE3FU5 141520123 IC50 = 34090 nM T83875 CKS8R1 141520127 IC50 = 109570 nM T83875 CX3DI7 141520133 IC50 > 200000 nM T83875 CUZ2C8 141766036 IC50 < 100 nM T83875 CA7H1W 141766041 IC50 = 230 nM T83875 CY3A7G 145948500 IC50 = 1.4 nM T83875 CKT3V1 145948504 IC50 = 1.9 nM T83875 CT48HM 145948506 IC50 = 20 nM T83875 C4C1JY 145948507 IC50 = 50 nM T83875 CM7FE5 145948508 IC50 = 7.4 nM T83875 CJ4Q9L 145948509 IC50 = 801 nM T83875 CHFL20 145948511 IC50 = 6 nM T83875 CEIL06 145948520 IC50 = 20 nM T83875 CQOP12 145948521 IC50 = 9 nM T83875 C71JXN 145948522 IC50 = 6.3 nM T83875 C8I4CY 145948524 IC50 = 140 nM T83875 C4C7VQ 145948525 IC50 = 34 nM T83875 CSR05F 145948530 IC50 = 18 nM T83875 CZJ2M5 145948531 IC50 = 2.3 nM T83875 C13EJK 145948532 IC50 = 1 nM T83875 CC2N4S 145948533 IC50 = 17 nM T83875 COL6M1 145948534 IC50 = 4.1 nM T83875 CJD26S 145948549 IC50 = 30 nM T83875 CZ61JB 145948550 IC50 = 3.9 nM T83875 C81KYR 145948553 IC50 = 6.3 nM T83875 CVF2R3 145948554 IC50 = 50 nM T83875 CD83FI 145948555 IC50 = 7.6 nM T83875 C7ID5T 145948556 IC50 = 65 nM T83875 CJ8PF4 145948559 IC50 = 13 nM T83875 C7IX0H 145948560 IC50 = 6.6 nM T83875 CK21IG 145948561 IC50 = 50 nM T83875 CW3CF1 145948562 IC50 = 14 nM T83875 C97JVF 145948622 IC50 > 30000 nM T83875 C9XO4M 145948655 IC50 > 30000 nM T83875 CHP2V5 145948690 IC50 > 30000 nM T83875 CLD12N 145949023 IC50 > 30000 nM T83875 C5GM0U 145949030 IC50 > 30000 nM T83875 CZ80NX 145949421 IC50 = 30200 nM T83875 C1TDL9 145949549 IC50 = 2660 nM T83875 CDA28I 145949712 IC50 = 21110 nM T83875 CM12NP 145949823 IC50 = 61338 nM T83875 C54UIF 145949921 IC50 = 6030 nM T83875 CRN6H7 145949934 IC50 = 8300 nM T83875 CPX50L 145949947 IC50 > 50000 nM T83875 CW3P6G 145950085 IC50 = 11200 nM T83875 CGQ3U6 145950141 IC50 = 9100 nM T83875 C81JWA 145950243 IC50 > 50000 nM T83875 CO2M5E 145950303 IC50 = 79700 nM T83875 C49AIV 145950338 IC50 = 4410 nM T83875 CRD3S7 145950766 IC50 = 3070 nM T83875 CT90WU 145950837 IC50 = 540 nM T83875 CC7Q3F 145950843 IC50 = 9003 nM T83875 C8SM2O 145950855 IC50 = 10 nM T83875 CX91AI 145950913 IC50 = 27200 nM T83875 C1VE0Q 145951053 IC50 = 2330 nM T83875 C8RQ2P 145951193 Ki = 6.6 nM T83875 CM3R8C 145951251 IC50 > 50000 nM T83875 C3U0WI 145951283 IC50 = 2060 nM T83875 CJN6H5 145951347 IC50 = 4330 nM T83875 CY91WG 145951519 IC50 > 50000 nM T83875 CAY7P0 145951540 IC50 > 50000 nM T83875 CO4X0H 145951870 IC50 = 10210 nM T83875 CX1P7H 145952331 IC50 > 100000 nM T83875 C8YD1P 145952456 IC50 = 42670 nM T83875 C19ZGF 145952532 IC50 = 4327 nM T83875 C47ABX 145952713 IC50 = 29100 nM T83875 CA0H2O 145952896 IC50 = 11393 nM T83875 C8LU9S 145953219 IC50 = 10559 nM T83875 CFE03V 145953575 IC50 > 60000 nM T83875 CCG6Z2 145953702 IC50 > 50000 nM T83875 CN47FR 145953732 IC50 = 64800 nM T83875 CJ1XM7 145953859 IC50 = 3690 nM T83875 CM3T6Y 145953870 IC50 = 9150 nM T83875 CRYS31 145954037 IC50 = 9020 nM T83875 CCV17M 145954104 IC50 = 1420 nM T83875 C1I9WM 145954115 IC50 = 15440 nM T83875 CUMJ40 145954156 IC50 = 103368 nM T83875 CL0XT8 145954248 IC50 = 39410 nM T83875 CC9A0N 145954291 IC50 = 1130 nM T83875 CUIY71 145954565 IC50 > 50000 nM T83875 CZ5MI9 145954575 IC50 > 50000 nM T83875 C3FS2N 145954793 IC50 = 65700 nM T83875 C8A4TF 145954923 IC50 > 60000 nM T83875 CVBH34 145954971 IC50 > 50000 nM T83875 C90TGE 145955059 IC50 > 60000 nM T83875 C8FSO7 145955146 IC50 > 60000 nM T83875 CE8G4I 145955186 IC50 = 20024 nM T83875 CZU84I 145955291 IC50 = 10393 nM T83875 CKU7Z5 145955423 IC50 = 7150 nM T83875 C37SYH 145955424 IC50 > 100000 nM T83875 CCZ2R9 145955785 IC50 = 10 nM T83875 CRTP17 145955809 IC50 > 60000 nM T83875 C2DF7C 145955811 IC50 = 7220 nM T83875 CQ6MY0 145956006 Ki = 4.4 nM T83875 C5XT4Z 145956132 IC50 > 100000 nM T83875 CHEG86 145956238 IC50 = 6330 nM T83875 CPY71F 145956290 IC50 > 100000 nM T83875 C4MUO0 145956291 IC50 = 4060 nM T83875 C2XOL5 145956393 IC50 > 50000 nM T83875 CDY0S5 145956567 IC50 = 470 nM T83875 C2D4LA 145956942 IC50 = 31200 nM T83875 C28IPH 145957131 IC50 = 1110 nM T83875 C0U5NS 145957329 IC50 = 7730 nM T83875 C9W6MV 145957333 IC50 = 1590 nM T83875 CGO4F6 145957401 IC50 = 10600 nM T83875 CJ03TU 145957740 IC50 = 50070 nM T83875 C9ES7D 145957769 IC50 = 45150 nM T83875 C4G3LT 145957957 IC50 = 31400 nM T83875 CN4R9J 145958017 IC50 > 60000 nM T83875 CY4EX0 145958214 IC50 = 7000 nM T83875 CUJQ65 145958271 IC50 = 1820 nM T83875 CC18RP 145958787 IC50 > 50000 nM T83875 CGD7Z3 145958889 IC50 = 3490 nM T83875 C93IGN 145958945 IC50 = 9550 nM T83875 C25OZA 145958966 IC50 = 15620 nM T83875 C5A1TY 145959187 IC50 > 60000 nM T83875 CZ1O7J 145959317 IC50 > 50000 nM T83875 C0M7PW 145959369 IC50 > 50000 nM T83875 CPF6B7 145959387 IC50 = 1770 nM T83875 C7DZA2 145959459 IC50 = 24300 nM T83875 C9FQH0 145959513 IC50 = 7800 nM T83875 CV8Z4N 145959672 IC50 = 3 nM T83875 CUXZ08 145959682 IC50 = 25583 nM T83875 CB6O5R 145959714 IC50 = 38000 nM T83875 C69BEI 145959843 IC50 = 85434 nM T83875 CYP62M 145959951 IC50 = 76200 nM T83875 CU58SO 145960091 IC50 > 60000 nM T83875 C37OHE 145960135 IC50 = 33800 nM T83875 CL0WE8 145960174 IC50 = 3990 nM T83875 C13WSY 145960214 IC50 = 10900 nM T83875 CG5KQ7 145960277 IC50 > 50000 nM T83875 C4V1GR 145960343 IC50 = 2560 nM T83875 C62JCL 145960933 IC50 > 10000 nM T83875 CFM39D 145962916 IC50 = 970 nM T83875 CD39PS 145963747 IC50 = 5200 nM T83875 CJ5DG6 145963998 IC50 = 67000 nM T83875 CQ5RX2 145964047 IC50 > 100000 nM T83875 C8E3AJ 145964075 IC50 > 100000 nM T83875 CF6Q8B 145964244 IC50 = 116370 nM T83875 C4KW1B 145964292 IC50 > 100000 nM T83875 CD2X4I 145964386 IC50 = 36000 nM T83875 CH5G8U 145964572 IC50 = 89350 nM T83875 CXJS15 145964929 IC50 > 100000 nM T83875 CZE6R5 145965009 IC50 > 30000 nM T83875 C9V4IH 145965010 IC50 = 56410 nM T83875 C2CL8F 145965108 IC50 = 59990 nM T83875 C7GF1E 145965278 IC50 = 54510 nM T83875 CLW9H6 145965317 IC50 = 53290 nM T83875 CVYM98 145965396 IC50 > 10000 nM T83875 CMYG28 145965829 IC50 > 10000 nM T83875 CTS35V 145966018 IC50 > 100000 nM T83875 CF06BV 145966566 IC50 = 5900 nM T83875 C7L0MY 145966586 IC50 = 71000 nM T83875 CAX84N 145966790 IC50 > 100000 nM T83875 CS5FC0 145966840 IC50 > 10000 nM T83875 C5D3HZ 145966917 IC50 > 10000 nM T83875 CB71YE 145966926 IC50 = 49170 nM T83875 CZES12 145967115 IC50 = 36870 nM T83875 C60ZBC 145967151 IC50 = 70020 nM T83875 CIRD04 145967411 IC50 > 100000 nM T83875 CIXR60 145967524 IC50 > 10000 nM T83875 CX9O3K 145967672 IC50 = 9900 nM T83875 C9Z3LA 145967889 IC50 = 9400 nM T83875 C03CRW 145968128 IC50 = 7100 nM T83875 CWJ64D 145968255 IC50 = 58000 nM T83875 CWX75L 145968655 IC50 = 7100 nM T83875 CXF29K 145968802 IC50 = 6900 nM T83875 CB80FD 145968869 IC50 = 15900 nM T83875 CV4H5D 145969277 IC50 = 11300 nM T83875 CQV1S7 145969296 IC50 > 100000 nM T83875 C9Z8WX 145969491 IC50 = 7900 nM T83875 C2FU9B 145969589 IC50 = 9900 nM T83875 CYMF27 145969637 IC50 > 10000 nM T83875 CSXF25 145969647 IC50 = 8200 nM T83875 CY32TF 145969707 IC50 = 9600 nM T83875 C0GWL4 145969718 IC50 = 15500 nM T83875 C6M2FZ 145970256 IC50 = 23000 nM T83875 C6A4SV 145970363 IC50 = 19900 nM T83875 C27EMD 145970504 IC50 > 100000 nM T83875 C67OFB 145970725 IC50 = 3400 nM T83875 C6PYZ0 145970731 IC50 = 19900 nM T83875 CW60FG 145970775 IC50 = 39000 nM T83875 C9IW2K 145970779 IC50 = 57500 nM T83875 C97VSH 145971024 IC50 = 9178 nM T83875 CZ5WB1 145971140 IC50 = 16600 nM T83875 C23KUV 145971152 IC50 = 8900 nM T83875 C6N7JF 145971479 IC50 = 53956 nM T83875 CVTO93 145971704 IC50 = 8180 nM T83875 C3Q1TN 145971772 IC50 > 60000 nM T83875 COE8K3 145971958 IC50 = 4860 nM T83875 CKY7V1 145971968 IC50 = 66317 nM T83875 CUTB21 145972060 IC50 > 10000 nM T83875 CQ7U1M 145972128 IC50 > 100000 nM T83875 C02NHL 145972143 IC50 > 10000 nM T83875 C19WJX 145972230 IC50 = 9330 nM T83875 CPNJ15 145972300 IC50 > 100000 nM T83875 CXIM57 145972351 IC50 = 94530 nM T83875 CO19QS 145972772 IC50 = 3275 nM T83875 CNE54W 145972804 IC50 > 10000 nM T83875 C6R8IL 145973192 IC50 = 13109 nM T83875 C5SM0J 145973231 IC50 = 11390 nM T83875 C1LM0W 145973337 IC50 = 72060 nM T83875 CP32EZ 145973435 IC50 = 93240 nM T83875 CE9JC0 145973764 IC50 = 38610 nM T83875 CAC9Q8 145973846 IC50 > 60000 nM T83875 CB5H6K 145973982 IC50 = 29260 nM T83875 C6F1WT 145974014 IC50 > 100000 nM T83875 C1I3SB 145974077 IC50 = 14611 nM T83875 CYSL73 145974355 IC50 = 6300 nM T83875 CY1G2F 145974565 IC50 = 36890 nM T83875 C1TI6B 145974586 IC50 > 10000 nM T83875 CFN8D6 145974596 IC50 > 100000 nM T83875 C8W2KY 145974736 IC50 = 70000 nM T83875 C9EFC7 145974855 IC50 > 100000 nM T83875 C1YRD3 145974906 IC50 = 55050 nM T83875 CU15SA 145974947 IC50 = 5514 nM T83875 C7O4SQ 145974973 IC50 = 4600 nM T83875 C3HPU6 145975029 IC50 = 24000 nM T83875 CO0D6E 145975284 IC50 = 69870 nM T83875 CR21PI 145975443 IC50 > 10000 nM T83875 C7NV3M 145975746 IC50 = 22700 nM T83875 C7CW4G 145975882 IC50 = 89500 nM T83875 CZO18H 145976060 IC50 = 77440 nM T83875 CR2MT1 145976177 IC50 > 10000 nM T83875 CZYI64 145976195 IC50 = 69150 nM T83875 CCG38X 145976354 IC50 = 40780 nM T83875 CDH04P 145977491 IC50 = 18790 nM T83875 C8IAL2 145977624 IC50 > 10000 nM T83875 CB53MH 145977978 IC50 = 78560 nM T83875 C9H1EZ 145978133 IC50 = 35400 nM T83875 C93MSO 145978282 IC50 > 100000 nM T83875 CB4RK0 145978554 IC50 = 24000 nM T83875 C1QE8L 145978587 IC50 > 10000 nM T83875 CQZ0G5 145978902 IC50 = 78200 nM T83875 CHX28E 145978908 IC50 = 80000 nM T83875 CHWP93 145979173 Ki = 40000 nM T83875 CJS5N8 145979426 IC50 = 88110 nM T83875 C4TR1C 145979433 IC50 = 4310 nM T83875 CQ30IN 145979533 Ki = 192840 nM T83875 C7HTX2 145979575 IC50 = 780 nM T83875 C15CDR 145979739 IC50 = 10990 nM T83875 CX2RW9 145979866 IC50 = 95200 nM T83875 C1D9ZU 145979972 IC50 = 72700 nM T83875 C0VAL8 145980562 IC50 = 100000 nM T83875 CW93VH 145980588 IC50 = 70500 nM T83875 CU0TA8 145980601 IC50 = 64500 nM T83875 CUI5C2 145980623 IC50 = 488.5 nM T83875 C87KIE 145981180 IC50 = 99080 nM T83875 CK0V8L 145981246 IC50 = 21600 nM T83875 CB9Q6H 145981331 IC50 = 65100 nM T83875 CN1RQ3 145981915 IC50 = 42500 nM T83875 CEM93S 145981925 IC50 = 109100 nM T83875 CX3M9J 145981988 IC50 = 38000 nM T83875 CG1BW6 145982188 IC50 = 62900 nM T83875 CS50XZ 145982212 IC50 = 73200 nM T83875 CWNB08 145982383 IC50 = 37800 nM T83875 CFNJ87 145982457 IC50 = 20500 nM T83875 CAC72J 145982690 IC50 = 69300 nM T83875 CG34HN 145983490 IC50 = 72520 nM T83875 C7VJ1L 145983695 IC50 = 46600 nM T83875 CV46GJ 145986363 Ki = 80 nM T83875 CW3RG1 145987055 IC50 = 205.5 nM T83875 C5A1VF 145987332 Ki = 19550 nM T83875 CYWE49 145987379 IC50 = 70600 nM T83875 C21BYI 145987407 IC50 > 100000 nM T83875 CVM40C 145987439 IC50 = 72100 nM T83875 CKV9T1 145987752 IC50 = 90200 nM T83875 C98DHT 145987800 IC50 = 52400 nM T83875 CA82TF 145987838 IC50 > 100000 nM T83875 C3M1ZO 145988042 IC50 = 39300 nM T83875 C0VRL2 145988393 IC50 = 17100 nM T83875 CVD20U 145988532 Ki = 57 nM T83875 C1XU7P 145988798 IC50 > 100000 nM T83875 CFQ97B 145989140 IC50 = 48400 nM T83875 CX5F4Z 145989197 IC50 = 160.5 nM T83875 CWJ1R2 145989205 IC50 = 60200 nM T83875 C2A8MY 145989254 IC50 = 93700 nM T83875 CUJ53A 145989396 IC50 = 310 nM T83875 C4C2IS 145989399 IC50 = 70900 nM T83875 CJFG45 145990271 IC50 = 27900 nM T83875 CSR71M 145990276 IC50 = 39100 nM T83875 CDIV28 145990279 IC50 = 94100 nM T83875 CDBW68 145990442 IC50 = 41500 nM T83875 CR59TZ 145990611 IC50 > 100000 nM T83875 CQ4R9F 145990749 IC50 = 62300 nM T83875 C5QZJ4 145990784 IC50 > 100000 nM T83875 C10HQC 145991026 IC50 > 100000 nM T83875 CO5V7B 145991298 IC50 = 64700 nM T83875 C70GLU 145991351 IC50 = 51640 nM T83875 C3Y7FC 145991399 IC50 = 72500 nM T83875 CKQ9N2 145991501 IC50 = 52900 nM T83875 CKU1A9 145991587 IC50 = 4910 nM T83875 C9L8FJ 145991954 IC50 = 70100 nM T83875 CRWN45 145992049 IC50 > 100000 nM T83875 C1O3VK 145992136 IC50 = 38100 nM T83875 CB9P8D 145992212 IC50 > 100000 nM T83875 C1WI3A 145992723 IC50 = 15300 nM T83875 CJ04DE 145992806 IC50 = 59600 nM T83875 C1JW3O 145992909 IC50 > 100000 nM T83875 CIH8O3 145993065 IC50 = 13400 nM T83875 CV4AT0 145993142 Ki = 26200 nM T83875 C5YMR4 145993208 IC50 > 100000 nM T83875 C3XT1C 145993229 IC50 = 41400 nM T83875 CUVC73 145993378 IC50 > 100000 nM T83875 CVY1T9 145993407 IC50 = 33420 nM T83875 CLST75 145993460 IC50 = 100000 nM T83875 C30CMY 145993498 IC50 > 100000 nM T83875 CYFO75 145993569 IC50 = 20370 nM T83875 CE0YD2 145993718 IC50 = 104300 nM T83875 CM0DW5 145993841 IC50 = 24700 nM T83875 CNY18A 145994134 IC50 > 100 nM T83875 CRQ31D 145994230 IC50 = 237 nM T83875 C4V2RJ 145994271 IC50 = 51300 nM T83875 CU9M1Y 145994293 IC50 = 58400 nM T83875 C4NZ6L 150525142 IC50 > 50000 nM T83875 CI32AF 150615303 IC50 = 12400 nM T83875 CF05TU 150717439 IC50 = 5243.7 nM T83875 CJE43S 150762943 IC50 = 17100 nM T83875 CJR07T 150914951 IC50 = 22500 nM T83875 C7E9LT 150956546 IC50 = 1570 nM T83875 CSDW79 151032063 IC50 = 5470 nM T83875 CP93LE 151074609 IC50 = 7370 nM T83875 CP8U5D 151566527 IC50 = 2310 nM T83875 C2U4KE 151661379 IC50 = 55500 nM T83875 CL8DP4 152061489 IC50 = 12000 nM T83875 CZFU85 152109514 IC50 = 1390 nM T83875 CN0ZQ9 152323773 IC50 = 168.8 nM T83875 C7D4UB 152687816 IC50 = 15800 nM T83875 CP56CH 152688549 IC50 = 751 nM T83875 CJY38R 153525743 IC50 > 50000 nM T83875 C2FUG3 153525745 IC50 = 300 nM T83875 CJM37F 153525746 IC50 = 4100 nM T83875 C5MCK8 153525747 IC50 = 2900 nM T83875 C2ZI9B 153525748 IC50 = 1100 nM T83875 C67IQJ 153525750 IC50 > 50000 nM T83875 CGP93O 153525752 IC50 = 3000 nM T83875 CS7F8Q 153525754 IC50 = 2200 nM T83875 C7U4GO 153525755 IC50 = 15900 nM T83875 CM97FW 153525756 IC50 = 4500 nM T83875 CQ4R8G 153525759 IC50 = 3200 nM T83875 CD81MP 153525760 IC50 = 8000 nM T83875 CS0ZN7 153525761 IC50 = 12400 nM T83875 CU16IY 153525763 IC50 = 140 nM T83875 C6ZDG0 153525764 IC50 = 13700 nM T83875 C02PQN 153525765 IC50 > 50000 nM T83875 CFR4W2 153525769 IC50 > 50000 nM T83875 CIVC40 153525771 IC50 = 10500 nM T83875 CD0J3R 153525775 IC50 > 50000 nM T83875 C1NK6C 153525776 IC50 = 200 nM T83875 CJ26VA 153525778 IC50 = 800 nM T83875 CS6N2Z 153525780 IC50 > 50000 nM T83875 CCI3U5 153525781 IC50 > 50000 nM T83875 CBV4E7 153525782 IC50 = 2700 nM T83875 CMJQ60 153525784 IC50 = 200 nM T83875 CM87OZ 153525785 IC50 > 50000 nM T83875 C6T9SI 153525786 IC50 > 50000 nM T83875 CVG27E 153525788 IC50 = 19200 nM T83875 C2YWN9 153525789 IC50 = 4400 nM T83875 CBC36V 153525792 IC50 = 18300 nM T83875 C8IW1V 153525795 IC50 = 2100 nM T83875 CFH9L5 153525796 IC50 = 28600 nM T83875 C52SJA 155510567 IC50 > 100000 nM T83875 CV02GT 155510689 IC50 = 24300 nM T83875 C9ATE6 155510755 IC50 = 31500 nM T83875 CB74UX 155510892 IC50 = 24060 nM T83875 CP5OS6 155511517 IC50 = 62800 nM T83875 C1NE6X 155511966 IC50 > 100000 nM T83875 C14FHM 155512092 IC50 > 50000 nM T83875 C54NIK 155512517 IC50 = 4550 nM T83875 CW6C3Q 155512810 IC50 = 39600 nM T83875 C2BGD3 155513276 IC50 = 79200 nM T83875 C21PXB 155513855 IC50 = 46200 nM T83875 CDLC76 155513877 IC50 = 1110 nM T83875 C9UT6Z 155513926 IC50 = 8120 nM T83875 CTQ3F4 155514293 IC50 = 56440 nM T83875 CRJ0A3 155514729 IC50 = 22100 nM T83875 C3VYW4 155514859 IC50 > 100000 nM T83875 C3HE8N 155515066 IC50 = 11700 nM T83875 CUI18M 155515157 IC50 = 55500 nM T83875 C3I9WB 155515459 IC50 = 9330 nM T83875 CR7C0G 155515606 IC50 = 490 nM T83875 C1F6GM 155515963 IC50 = 12460 nM T83875 CNV02U 155516016 IC50 > 10000 nM T83875 C7BF6M 155516327 IC50 = 24700 nM T83875 CPBN03 155516779 IC50 = 810 nM T83875 CAQ9G2 155516780 IC50 = 540 nM T83875 C5QJ4R 155516939 IC50 > 10000 nM T83875 CEA8D5 155516976 IC50 > 100000 nM T83875 C0N9ZD 155517085 IC50 = 46121.5 nM T83875 CTE5N3 155517491 IC50 > 500000 nM T83875 CUAG18 155517670 IC50 = 14700 nM T83875 C5PO3X 155517932 IC50 > 500000 nM T83875 C8JMD2 155518028 IC50 = 26100 nM T83875 C2CWD9 155518118 IC50 = 23190 nM T83875 CIM31H 155518405 IC50 = 20300 nM T83875 CKC0J2 155518449 IC50 > 500000 nM T83875 CHQX97 155518786 IC50 = 822 nM T83875 CW7TP1 155519024 IC50 > 100000 nM T83875 C36LGV 155519027 IC50 = 12890 nM T83875 CR9ZW6 155519043 IC50 = 980 nM T83875 CP8UD6 155520012 IC50 = 19700 nM T83875 C3B0WM 155520213 IC50 > 100000 nM T83875 C76VBO 155520546 IC50 = 28550 nM T83875 CY25CV 155520663 IC50 > 10000 nM T83875 C7R8UB 155520744 IC50 > 10000 nM T83875 CLN8H5 155520953 IC50 = 1100 nM T83875 C3DZQ4 155521124 IC50 = 68.4 nM T83875 CF28LO 155521322 IC50 = 24990 nM T83875 CP0E2K 155521356 IC50 = 1900 nM T83875 C86WXD 155521569 IC50 = 16600 nM T83875 CPM03G 155521729 IC50 > 10000 nM T83875 CEAV65 155521960 IC50 = 2770 nM T83875 C4YPF9 155522024 IC50 > 50000 nM T83875 CLK83G 155522136 IC50 = 34150 nM T83875 C4F7XP 155522484 IC50 = 43100 nM T83875 CB57GS 155522741 IC50 = 68000 nM T83875 C8ZOV5 155522894 IC50 > 100000 nM T83875 CTH80O 155523061 IC50 = 63900 nM T83875 CKR9P2 155523992 IC50 = 10500 nM T83875 C0JDC4 155524002 IC50 > 100000 nM T83875 C7STO9 155524244 IC50 = 1590 nM T83875 CED31W 155524277 IC50 = 4510 nM T83875 CS1LG9 155525089 IC50 > 100000 nM T83875 CI0V5F 155525579 IC50 > 100000 nM T83875 C2YS9O 155525759 IC50 = 2810 nM T83875 C7IQ6J 155525760 IC50 = 2300 nM T83875 CT4XV9 155525799 IC50 = 26100 nM T83875 CQU8C1 155526013 IC50 > 500000 nM T83875 CKA2M3 155526429 IC50 = 230 nM T83875 C9Q0OP 155526667 IC50 = 21140 nM T83875 CY0P1G 155527083 IC50 > 500000 nM T83875 C2UO1C 155527178 IC50 > 500000 nM T83875 CLF6J9 155527441 IC50 > 100000 nM T83875 C5Q1LN 155528022 IC50 = 116800 nM T83875 CCU17Y 155528388 IC50 = 21200 nM T83875 CCA76W 155528448 IC50 > 50000 nM T83875 CK37ZL 155528508 IC50 = 85200 nM T83875 CPU41A 155528785 IC50 = 91400 nM T83875 CQM2L6 155529262 IC50 > 50000 nM T83875 C0Q8PH 155529386 IC50 = 858 nM T83875 CGX6S4 155529530 IC50 > 10000 nM T83875 CM9E2L 155529630 IC50 > 200000 nM T83875 CDT04B 155529889 IC50 > 100000 nM T83875 CPOR92 155530007 IC50 = 53120 nM T83875 CR3C2A 155530056 IC50 > 500000 nM T83875 C34VYA 155530298 IC50 > 10000 nM T83875 CF4JS0 155530576 IC50 = 62200 nM T83875 C2YDZ8 155531112 IC50 > 10000 nM T83875 C5X1QC 155531135 IC50 > 10000 nM T83875 CS35DE 155531420 IC50 > 100000 nM T83875 CI0XL3 155531445 IC50 = 23900 nM T83875 CO1B6G 155531477 IC50 = 13600 nM T83875 C92HMB 155532012 IC50 > 10000 nM T83875 CD14WR 155532205 IC50 = 870 nM T83875 CYL4B2 155532320 IC50 = 11000 nM T83875 CXMC14 155532373 IC50 > 10000 nM T83875 C03YPC 155532460 IC50 = 24700 nM T83875 CD73OS 155532519 IC50 = 136100 nM T83875 CMKP85 155532627 IC50 > 50000 nM T83875 CMZ3F5 155533066 IC50 = 234600 nM T83875 CBL16Y 155533456 IC50 = 3500 nM T83875 C8FCH7 155533611 IC50 > 10000 nM T83875 C9WO1Z 155533882 IC50 > 10000 nM T83875 CYN5O8 155534304 IC50 = 550 nM T83875 CV5TY2 155535062 IC50 = 89330 nM T83875 CZV42I 155535793 IC50 = 25830 nM T83875 CA1S4K 155535904 IC50 = 2410 nM T83875 C0OGM5 155536279 IC50 = 12400 nM T83875 CH7C5J 155536981 IC50 > 100000 nM T83875 CMG75B 155537001 IC50 > 10000 nM T83875 C8ZG7F 155537023 IC50 > 10000 nM T83875 CS9M4P 155537529 IC50 = 1290 nM T83875 CV39TC 155537638 IC50 = 24600 nM T83875 CUI68E 155538243 IC50 > 500000 nM T83875 C87THM 155538450 IC50 = 88300 nM T83875 C1BHZ0 155538647 IC50 = 310900 nM T83875 CB6W7X 155538837 IC50 = 61500 nM T83875 C54MIG 155539279 IC50 = 32060 nM T83875 CME98X 155539363 IC50 = 4240 nM T83875 CF6ZE5 155540615 IC50 > 10000 nM T83875 C3P1ZT 155540839 IC50 > 1000 nM T83875 CJ2G7I 155540870 IC50 < 300000 nM T83875 C2L9TS 155540948 IC50 > 1000 nM T83875 C83BZU 155540992 IC50 > 100000 nM T83875 CBE65T 155541185 IC50 > 10000 nM T83875 C19HQM 155541262 IC50 > 1000 nM T83875 C7XBV5 155542241 IC50 = 18200 nM T83875 C4KWU5 155542251 IC50 > 100000 nM T83875 CX4P8S 155542351 IC50 = 4100 nM T83875 CCV87Q 155542600 IC50 > 1000 nM T83875 C8JY0G 155542643 IC50 > 100000 nM T83875 C0H7IT 155542980 IC50 = 2680 nM T83875 C9VS1J 155543043 IC50 = 267400 nM T83875 CMU24O 155543147 IC50 = 108200 nM T83875 CQB52M 155543548 IC50 = 55900 nM T83875 CB1XH5 155544104 IC50 = 8270 nM T83875 CZ8KL6 155544230 IC50 = 134700 nM T83875 CPXY64 155544313 IC50 = 50000 nM T83875 C5AE8I 155544346 IC50 = 39740 nM T83875 C5HDZ9 155544380 IC50 = 210 nM T83875 C5Y4BH 155545414 IC50 > 10000 nM T83875 C7JNP0 155545476 IC50 = 56230 nM T83875 CLB1P9 155545663 IC50 = 3900 nM T83875 C7RWG6 155545712 IC50 = 553500 nM T83875 CP15TU 155546048 IC50 > 100000 nM T83875 C4BHE8 155546183 IC50 > 1000 nM T83875 CF4V6H 155546226 IC50 > 100000 nM T83875 C1X2GS 155546843 IC50 > 10000 nM T83875 C60OKG 155547117 IC50 = 40860 nM T83875 C0MYF3 155547509 IC50 = 80305.3 nM T83875 CK1X5S 155547588 IC50 > 1000 nM T83875 C8Q7JG 155547782 IC50 > 1000 nM T83875 C12EGC 155547881 IC50 = 13600 nM T83875 C0OAH3 155547969 IC50 = 83800 nM T83875 C4MIT2 155548780 IC50 > 1000 nM T83875 CON2H6 155548824 IC50 = 25570 nM T83875 CW89KS 155549035 IC50 = 1100 nM T83875 CUK96G 155549201 IC50 = 26100 nM T83875 C3M2DC 155549619 IC50 = 47000 nM T83875 CG9K3X 155549681 IC50 = 56100 nM T83875 CY5P6K 155549919 IC50 = 94297 nM T83875 C7ARS4 155550007 IC50 = 700 nM T83875 CC45SE 155550088 IC50 > 1000 nM T83875 C7ZK8C 155550291 IC50 = 173400 nM T83875 C2IU1J 155550532 IC50 > 1000 nM T83875 CWL16Z 155550534 IC50 > 100000 nM T83875 CVUZ30 155550746 IC50 = 26100 nM T83875 C9CKH4 155550772 IC50 = 60 nM T83875 CM41NQ 155550778 IC50 > 100000 nM T83875 C1J7SD 155550841 IC50 = 3590 nM T83875 CEF57Y 155551313 IC50 = 38400 nM T83875 COR5T3 155551621 IC50 > 200000 nM T83875 C8JD0O 155551671 IC50 = 9190 nM T83875 CCD10R 155551712 IC50 > 100000 nM T83875 CI0WL8 155551843 IC50 = 726.1 nM T83875 C5H0FB 155552050 IC50 > 500000 nM T83875 CA3SR7 155552282 IC50 = 22020 nM T83875 CFZ7K1 155552358 IC50 = 155150 nM T83875 CM40UT 155552539 IC50 > 100000 nM T83875 CIQH30 155552719 IC50 > 1000 nM T83875 CT9D2Y 155553307 IC50 = 118844.3 nM T83875 C1RLI0 155553370 IC50 > 100000 nM T83875 C1A5OR 155553697 IC50 > 10000 nM T83875 CF1CQ9 155553798 IC50 = 3000 nM T83875 CC98IO 155554016 IC50 = 1110 nM T83875 CR2YV5 155554100 IC50 = 91200 nM T83875 CP10LB 155554293 IC50 > 500000 nM T83875 CSI9P4 155554561 IC50 > 100000 nM T83875 CT06QZ 155555033 IC50 = 1700 nM T83875 CQ4X0Z 155555067 IC50 = 94300 nM T83875 CQKH19 155555069 IC50 = 8570 nM T83875 CCV7X8 155555111 IC50 = 436500 nM T83875 C57MKC 155555241 IC50 > 1000 nM T83875 CQK21Y 155555466 IC50 = 2200 nM T83875 CR97GM 155555497 IC50 > 500000 nM T83875 CXMC57 155555780 IC50 = 7500 nM T83875 CJ73SL 155556032 IC50 > 1000 nM T83875 C8UQR0 155556261 IC50 = 2600 nM T83875 CJ75TC 155556370 IC50 > 50000 nM T83875 CV9P2M 155556457 IC50 > 10000 nM T83875 CC14ON 155556524 IC50 > 1000 nM T83875 CSN6O4 155556536 IC50 > 100000 nM T83875 C8QW7M 155556988 IC50 > 10000 nM T83875 CGZ08K 155557025 IC50 = 17300 nM T83875 C9FG2V 155557097 IC50 = 1720 nM T83875 CTVQ18 155557424 IC50 = 20990 nM T83875 CJ16GB 155557960 IC50 > 1000 nM T83875 C4I5JH 155558217 IC50 > 500000 nM T83875 C0W7AL 155558312 IC50 > 10000 nM T83875 CE4B5Q 155558687 IC50 = 2370 nM T83875 C9XQ0B 155559130 IC50 = 2240 nM T83875 CTI57G 155559203 IC50 > 100000 nM T83875 CP87XK 155559423 IC50 > 1000 nM T83875 CXU9Q2 155559464 IC50 = 3013.7 nM T83875 C0AI5O 155560069 IC50 = 1960 nM T83875 C2KI9B 155560090 IC50 = 7398.7 nM T83875 CP3T1Z 155560136 IC50 > 500000 nM T83875 C1H2BO 155560312 IC50 > 50000 nM T83875 C8B7CG 155560391 IC50 > 1000 nM T83875 C3OP1F 155560545 IC50 > 1000 nM T83875 C51KNM 155560680 IC50 = 24930 nM T83875 CXJ23G 155560844 IC50 > 100000 nM T83875 CU0E7C 155561006 IC50 > 100000 nM T83875 C2BH3L 155561208 IC50 > 200000 nM T83875 C6P9GA 155561569 IC50 = 1400 nM T83875 C1IA4X 155561597 IC50 > 10000 nM T83875 C5R3LT 155561606 IC50 = 2230 nM T83875 CWAG35 155561892 IC50 = 19800 nM T83875 C2JQ3C 155561938 IC50 > 50000 nM T83875 CK5G2U 155562162 IC50 = 10100 nM T83875 CUK35V 155562664 IC50 = 12180 nM T83875 C1NF2M 155562789 IC50 > 100000 nM T83875 C9JPF8 155563044 IC50 > 500000 nM T83875 CM46KC 155563177 IC50 > 1000 nM T83875 CQ19VC 155563189 IC50 > 1000 nM T83875 CA27NL 155563199 IC50 > 10000 nM T83875 CWBO72 155563250 Ki = 140 nM T83875 CS85JQ 155563497 IC50 = 41100 nM T83875 C26SAU 155563561 IC50 = 30100 nM T83875 CPTM25 155563673 IC50 > 100000 nM T83875 C2IGH8 155563922 IC50 = 29800 nM T83875 CZ6PB4 155564063 IC50 = 79455 nM T83875 COF96P 155564105 IC50 > 100000 nM T83875 CE2V5Y 155564179 IC50 > 1000 nM T83875 CY6OR7 155564797 IC50 = 1200 nM T83875 C83BSZ 155564858 IC50 > 500000 nM T83875 CUA4I7 155565084 IC50 = 2100 nM T83875 CVY9L7 155565232 IC50 = 34400 nM T83875 CKGC67 155565439 IC50 > 10000 nM T83875 C8N3PQ 155565636 IC50 > 1000 nM T83875 C8OL6E 155567040 IC50 = 10610 nM T83875 C9Q7WZ 155567401 IC50 > 200000 nM T83875 C7GU2Y 155568113 IC50 = 252200 nM T83875 CUT84A 155568798 IC50 > 100000 nM T83875 C3X5ML 155568799 IC50 = 18940 nM T83875 C8S0FZ 155568919 IC50 = 20790 nM T83875 CQ1LV7 135508617 IC50 = 236 nM T83875 CGK7B1 135511529 IC50 = 12167 nM T83875 CRKP76 136016509 IC50 = 8000 nM T83875 D00AVR 135476741 IC50 = 35 nM T83875 D00JUD 184462 IC50 = 7240 nM T83875 D00KDZ 44588139 Ki = 10000000 nM T83875 D00OLX 46232855 Ki = 180 nM T83875 D00OQL 3852139 IC50 = 235 nM T83875 D00RIX 5280443 IC50 = 1550 nM T83875 D00RNZ 910172 IC50 = 3490 nM T83875 D00WSM 599289 IC50 = 14500 nM T83875 D00WVG 584447 IC50 = 7883 nM T83875 D01LUB 4297278 IC50 = 400 nM T83875 D01PES 20037787 Ki = 100000000 nM T83875 D02AQM 6918822 IC50 = 57000 nM T83875 D02FJX 46232854 Ki = 51 nM T83875 D02ZZA 44424447 Ki = 75 nM T83875 D03EPY 7046 Ki = 210000 nM T83875 D03KDD 10464479 Ki = 5395106.23 nM T83875 D03LGV 11241513 IC50 = 1600 nM T83875 D03PXS 341782 IC50 = 13120 nM T83875 D04DYO 5281666 IC50 = 190 nM T83875 D04FLL 20242416 Ki > 100000 nM T83875 D04LPY 46232853 Ki = 180 nM T83875 D04TZI 12098585 IC50 = 65000 nM T83875 D05ANK 44588172 Ki = 59979107.63 nM T83875 D05CCT 4139 IC50 = 70 nM T83875 D05HJT 869109 IC50 = 15980 nM T83875 D05ODW 91510 IC50 = 85800 nM T83875 D05OXR 12209843 Ki = 100000000 nM T83875 D05QOR 5280460 IC50 > 20000 nM T83875 D05WQN 46400456 Ki = 18290 nM T83875 D05ZUX 44207909 Ki >= 1000 nM T83875 D06AAA 11390419 IC50 = 89000 nM T83875 D06AJP 44575103 Ki = 5600 nM T83875 D07BAO 5289289 Ki = 1900 nM T83875 D07GUX 42629116 Ki = 717 nM T83875 D07LCU 27647057 Ki = 5000345.35 nM T83875 D07NBB 46232852 Ki = 23 nM T83875 D07ULQ 11008237 Ki = 74989420.93 nM T83875 D07WFU 44577750 IC50 = 10000 nM T83875 D08CNS 3748 IC50 = 837 nM T83875 D08FFH 701943 IC50 = 3.78 nM T83875 D08FXH 46233267 Ki = 6620 nM T83875 D08HNJ 44588136 Ki = 454988060.2 nM T83875 D08ILX 24219274 Ki = 39450 nM T83875 D08NQM 5289247 IC50 = 165800 nM T83875 D08PEW 44588208 Ki = 100000000 nM T83875 D08PHY 11171752 IC50 = 3600 nM T83875 D08QZP 13680885 Ki = 476430986.8 nM T83875 D08SSS 44424448 Ki = 30 nM T83875 D08TFN 4996817 Ki = 16200 nM T83875 D08YCE 46232851 Ki = 36 nM T83875 D09HBX 10374615 IC50 = 12000 nM T83875 D09NNZ 46947643 Ki = 2580 nM T83875 D09XSB 42628986 Ki = 61 nM T83875 D0A1CM 5281855 EC50 = 1600 nM T83875 D0A1RE 44407281 IC50 = 40.5 nM T83875 D0A2AF 5289295 Ki = 4900 nM T83875 D0A4FA 11019886 Ki = 250034536.2 nM T83875 D0A4IY 5196 IC50 = 6700 nM T83875 D0B1WD 724200 IC50 = 15670 nM T83875 D0B6MV 658198 Ki = 340 nM T83875 D0C1LI 53378764 IC50 = 0.27 nM T83875 D0C8RD 11085165 Ki = 599791076.3 nM T83875 D0C9WW 16750123 Ki = 11000 nM T83875 D0D5KD 46233198 Ki = 60000 nM T83875 D0D6OR 46233269 Ki > 100000 nM T83875 D0D6QI 24219273 Ki = 8180 nM T83875 D0DQ6Z 8530 Ki = 7700 nM T83875 D0E4HB 8443728 IC50 = 48351 nM T83875 D0E8IE 3110315 IC50 = 9970 nM T83875 D0F2DC 11816512 IC50 = 13000 nM T83875 D0F7JK 821483 Ki = 3499451.67 nM T83875 D0F7KG 2329349 IC50 = 6880 nM T83875 D0GN5Z 5281295 IC50 = 4160 nM T83875 D0H0GZ 599290 IC50 = 19450 nM T83875 D0H1VT 11423691 IC50 = 18000 nM T83875 D0H5MV 16110305 Ki = 230144181.7 nM T83875 D0HU4J 5004199 Ki > 100000 nM T83875 D0I2GP 50876172 IC50 = 23731 nM T83875 D0I3XA 6422124 IC50 = 11000 nM T83875 D0IA3U 44442376 IC50 = 644 nM T83875 D0ID3Y 46233197 Ki > 100000 nM T83875 D0J0QW 46233266 Ki = 9600 nM T83875 D0J2UA 135433933 IC50 = 5.6 nM T83875 D0JN9R 223566 Ki = 590 nM T83875 D0K5LJ 5289310 IC50 = 17700 nM T83875 D0K9UN 589138 Ki = 130016957.8 nM T83875 D0KB2R 42776886 Ki = 10000000 nM T83875 D0KU2D 899774 Ki = 399944749.8 nM T83875 D0LI3J 3080926 Ki = 17000 nM T83875 D0M2EM 4650 IC50 = 4820 nM T83875 D0M4GR 46233264 Ki = 10000 nM T83875 D0M7BR 5280378 IC50 = 31200 nM T83875 D0M8UY 72139 IC50 = 9770 nM T83875 D0MO1O 11805737 Ki = 285759054.3 nM T83875 D0N8UE 16110292 Ki = 19998618.7 nM T83875 D0NS1S 5280442 Ki = 59.2 nM T83875 D0O0QN 11492774 IC50 = 12350 nM T83875 D0O2UK 413448 Ki = 349945167 nM T83875 D0P3DV 16110290 Ki = 54954087.39 nM T83875 D0P4GF 25139469 IC50 = 2380 nM T83875 D0Q1IP 5273551 IC50 = 14791.08 nM T83875 D0Q2QA 44424446 Ki = 133 nM T83875 D0R4PR 11623661 IC50 = 5310 nM T83875 D0R6FJ 64961 Ki = 260 nM T83875 D0S0JH 44563082 IC50 = 12200 nM T83875 D0SN3L 16110286 Ki = 419758984 nM T83875 D0SP2O 7054 Ki = 5940 nM T83875 D0T2RY 9948320 Ki >= 1000 nM T83875 D0T3XC 46233268 Ki = 2500 nM T83875 D0T3ZS 46233265 Ki > 100000 nM T83875 D0T9ZL 2703 Ki = 220 nM T83875 D0TL3S 25139473 IC50 = 11930 nM T83875 D0TU7I 5353365 IC50 > 10000 nM T83875 D0U9VX 11708692 IC50 = 2510 nM T83875 D0UL6Y 11401479 IC50 = 270000 nM T83875 D0V0TN 23020609 Ki = 69984199.6 nM T83875 D0V3NT 34521 IC50 = 980 nM T83875 D0V6DF 11615193 IC50 = 1300 nM T83875 D0X8HH 44575104 Ki = 2200 nM T83875 D0X8RN 6971118 IC50 = 11000 nM T83875 D0XJ7I 6683 Ki = 422 nM T83875 D0Y0LQ 44588174 Ki = 625172692.8 nM T83875 D0Y1XS 701990 IC50 = 2560 nM T83875 D0Y4JQ 16110288 Ki = 699841996 nM T83875 D0Y4SO 46223113 IC50 > 150000 nM T83875 D0Y7HG 5281616 IC50 = 130 nM T83875 D0Y8AN 5195 IC50 = 67250 nM T83875 D0YO7C 12627221 Ki = 169824365.3 nM T83875 D0Z0ZU 23661626 Ki = 22 nM T83875 D0Z5BU 46233199 Ki = 40000 nM T83875 D0Z5YO 8023988 Ki = 29991625.19 nM T25258 D00AXJ 4189 IC50 = 2000 nM T25258 D00KHM 16362 IC50 = 800 nM T25258 D00YZD 54726191 IC50 > 90000 nM T25258 D01XNB 4594 IC50 = 97200 nM T25258 D01ZII 2726 Ki = 600 nM T25258 D02DPA 2756 IC50 > 50000 nM T25258 D02OZE 2724385 IC50 > 50000 nM T25258 D02YIZ 12560 IC50 = 43000 nM T25258 D03DDR 3034034 IC50 = 1700 nM T25258 D03IGH 213039 IC50 = 6600 nM T25258 D04JEE 4946 Ki = 48000 nM T25258 D04LVK 57379345 EC50 = 89 nM T25258 D04XVN 11707110 EC50 = 247 nM T25258 D05NOS 5568 Ki = 15700 nM T25258 D07BSQ 5994 IC50 = 48977.88 nM T25258 D07IQS 148192 IC50 = 67800 nM T25258 D07KSG 2733526 Ki = 100 nM T25258 D07POC 176870 IC50 = 26000 nM T25258 D09DHY 6167 IC50 > 50000 nM T25258 D09GOS 2812 IC50 = 6700 nM T25258 D0A0OO 65016 IC50 > 100000 nM T25258 D0A4IJ 441300 IC50 > 500000 nM T25258 D0AZ3C 5291 IC50 = 7244.36 nM T25258 D0B7EB 36462 IC50 > 50000 nM T25258 D0BP9C 193962 IC50 = 7600 nM T25258 D0C4RB 36314 IC50 = 2596 nM T25258 D0D1AL 3559 Ki = 200 nM T25258 D0H3HM 60795 IC50 = 780 nM T25258 D0I2MK 4171 Ki = 200000 nM T25258 D0IT2G 5743 IC50 > 50000 nM T25258 D0J2KV 4932 EC50 = 320 nM T25258 D0J4JM 5770 Ki = 100 nM T25258 D0KR5B 5754 IC50 > 50000 nM T25258 D0L5WM 2157 Ki = 3200 nM T25258 D0NS6H 3152 IC50 = 34850 nM T25258 D0O5NK 65028 IC50 = 1300000 nM T25258 D0OB1J 39186 IC50 = 42657.95 nM T25258 D0R0FE 2520 IC50 = 4.9 nM T25258 D0R1RS 3715 IC50 = 28000 nM T25258 D0R3JB 4212 IC50 = 1501 nM T25258 D0R4OM 5566 Ki = 6500 nM T25258 D0T0KA 4474 IC50 = 950 nM T25258 D0U5GB 92727 IC50 = 10300 nM T25258 D0U6LM 4192 IC50 > 50000 nM T25258 D0V7CF 5362440 IC50 > 100000 nM T25258 D0W9MM 13342 Ki = 100 nM T25258 D0WE3O 5288826 IC50 > 50000 nM T25258 D0WI3T 441243 IC50 = 1600 nM T25258 D0ZU9R 392622 IC50 = 12000 nM T25258 D01GFX 11640390 EC50 = 2090 nM T25258 D02QWY 24785538 IC50 = 17700 nM T25258 D0CE0O 11513676 IC50 = 590 nM T25258 D0D2TZ 11303106 IC50 = 700 nM T25258 D0G7UX 5284373 EC50 = 32 nM T25258 D0U2BH 65064 IC50 = 124.1 nM T25258 D0U3EP 445154 IC50 = 60000 nM T25258 D0W8XT 60663 IC50 = 1500 nM T25258 D0O2EF 56946615 IC50 = 2000 nM T25258 D0V7UQ 56946834 IC50 = 2600 nM T25258 D03ISE 71144 Ki = 5500 nM T25258 D04RLX 148201 IC50 = 0.66 nM T25258 D06DCL 153997 IC50 = 3490 nM T25258 D07FJM 5743186 IC50 = 24100 nM T25258 D08SOF 5405 IC50 = 1100 nM T25258 D09FGX 119373 EC50 = 2000 nM T25258 D09TGX 5281884 IC50 = 501.19 nM T25258 D0B1MJ 6918097 EC50 = 60 nM T25258 D0OS6O 60149 IC50 = 6500 nM T25258 D0SR4G 6450807 IC50 = 31.62 nM T25258 D0T3ME 156422 EC50 = 524 nM T25258 D0Y2HR 2247 IC50 = 300 nM T25258 C52MFS 1756 EC50 > 100000 nM T25258 C0H8GR 3191 IC50 = 1500 nM T25258 CY4WG9 3793 IC50 = 2100 nM T25258 C9LCD8 3823 IC50 = 1000 nM T25258 C93BJO 5039 IC50 > 50000 nM T25258 CV24FH 10228 IC50 = 34000 nM T25258 C7H2NQ 21138 IC50 = 583000 nM T25258 CGKI54 22673 EC50 = 76400 nM T25258 C46BVP 46163 EC50 = 9073 nM T25258 C7CTS4 46186 EC50 = 3197 nM T25258 CY7DJ0 46199 EC50 = 128000 nM T25258 C28VFY 60602 IC50 = 707.95 nM T25258 CP8F7B 64143 IC50 = 1700 nM T25258 CJ3QB0 65218 Ki = 100 nM T25258 CA02CO 65808 Ki = 1600 nM T25258 CQ9MW6 68077 IC50 = 39000 nM T25258 C8C1JP 72343 IC50 = 1.59 nM T25258 CB6G3Z 91536 Ki = 170000 nM T25258 C0QET9 91773 IC50 = 21500 nM T25258 C1CWL8 92305 IC50 = 2090 nM T25258 C5ZCH7 97332 IC50 = 23400 nM T25258 CL97OF 97548 IC50 = 19700 nM T25258 C6I9HU 97860 IC50 = 64000 nM T25258 CZB67X 98608 IC50 = 32000 nM T25258 C52FVK 104972 IC50 = 4240 nM T25258 CTV78S 105010 IC50 = 44300 nM T25258 C09TNA 107927 EC50 = 3021 nM T25258 CY5Q6I 117804 EC50 > 500000 nM T25258 CZ8S4F 133055 IC50 = 4800 nM T25258 CV03LW 133129 IC50 = 170 nM T25258 C8NLJ2 145659 IC50 = 29000 nM T25258 C4FEY6 147157 IC50 = 15000 nM T25258 C7E5NC 150893 IC50 = 31000 nM T25258 CM23KQ 154172 EC50 = 6310 nM T25258 C3O4NA 179651 IC50 = 19140 nM T25258 CBA92W 183463 IC50 = 100400 nM T25258 CA3NK8 193841 EC50 = 28300 nM T25258 CR67FB 243037 EC50 > 100000 nM T25258 CABJ72 276138 IC50 = 4000 nM T25258 CHCP41 279081 IC50 = 15380 nM T25258 CN8ZL4 298546 EC50 = 53000 nM T25258 CP5B4K 369597 IC50 = 29000 nM T25258 CLD6J9 441074 IC50 = 2200 nM T25258 CWX96E 443274 EC50 = 1020 nM T25258 C1KVC4 443939 IC50 = 96910 nM T25258 CU1OM0 507272 IC50 = 3800 nM T25258 CZN1R3 507273 IC50 < 1000 nM T25258 C3J7OT 507274 IC50 = 6100 nM T25258 COI2C9 560674 EC50 > 100000 nM T25258 C0BZF7 639630 EC50 = 272500 nM T25258 CKT0V3 647240 IC50 > 200000 nM T25258 C0ZNP7 658081 EC50 = 2240 nM T25258 CTF2J0 687260 EC50 > 100000 nM T25258 CF3Q9N 703068 EC50 = 970 nM T25258 CO3TV1 704281 EC50 = 900 nM T25258 CNS78D 719277 IC50 = 3000 nM T25258 CUJ25K 721094 EC50 = 4590 nM T25258 CWU41X 750967 EC50 = 1310 nM T25258 C8OB6U 787509 IC50 = 4780 nM T25258 CBG3A2 914453 EC50 = 5940 nM T25258 CKZG90 921146 EC50 = 4150 nM T25258 C7D1QN 921567 EC50 > 100000 nM T25258 CK8TP4 1019287 IC50 = 20000 nM T25258 CWZ3L5 1087479 EC50 = 640 nM T25258 CL5WY4 1212338 EC50 = 1310 nM T25258 C3ZRH1 1221769 EC50 > 500000 nM T25258 CV7F8O 1418188 IC50 = 6370 nM T25258 CFJ6N3 1563361 EC50 = 311800 nM T25258 CB4GE0 1596119 EC50 = 3500 nM T25258 C4PU0N 1745958 EC50 = 17700 nM T25258 CQT4J5 2094802 IC50 > 100000 nM T25258 CX95WT 2270285 EC50 = 2650 nM T25258 C1A0FV 2298706 IC50 = 6800 nM T25258 C2ZDU4 2562583 IC50 = 12380 nM T25258 C2YC8B 2729881 IC50 = 15500 nM T25258 CW6SA0 2787558 IC50 > 100000 nM T25258 C7V3AY 2856734 EC50 = 599 nM T25258 CB1UT8 2856987 EC50 = 907 nM T25258 C57FZH 2926848 EC50 = 730 nM T25258 C4I1VF 2950589 IC50 = 2180 nM T25258 CX73PS 2951338 IC50 = 5320 nM T25258 CVX35C 2968016 EC50 = 207000 nM T25258 C63ANR 2968321 EC50 = 2087 nM T25258 CQ65MR 2968485 EC50 = 31960 nM T25258 CLGO78 2979948 IC50 = 500 nM T25258 C01JRM 3034694 IC50 = 15000 nM T25258 C85MYW 3036703 IC50 = 58.88 nM T25258 CQT28C 3112056 EC50 = 25130 nM T25258 CQ5G2S 3115657 EC50 > 100000 nM T25258 C9JUX7 3117509 EC50 = 760 nM T25258 C4N1DX 3117511 EC50 = 290 nM T25258 CWA3Z9 3120483 EC50 = 1210 nM T25258 CV85QH 3464805 EC50 = 640 nM T25258 C7Y1VG 3474421 EC50 = 302100 nM T25258 C70HAY 3619040 EC50 = 97 nM T25258 CD9G4Z 3621388 EC50 > 20000 nM T25258 CGXJ91 3632476 EC50 = 49000 nM T25258 C3YKU9 3639226 EC50 = 110 nM T25258 C41OWQ 3734747 EC50 = 460 nM T25258 C78KSM 3906724 EC50 > 50000 nM T25258 C2EDO0 3988866 EC50 = 20930 nM T25258 C72VLI 4022553 IC50 = 7940 nM T25258 C16FRV 4185749 EC50 = 280 nM T25258 CQ3G2Y 4363326 EC50 = 1000 nM T25258 CKGZ01 4447723 EC50 = 11890 nM T25258 CN3ZY9 4594014 EC50 > 100000 nM T25258 CHV3N6 4786429 IC50 = 14700 nM T25258 CKG0Q7 4839583 IC50 = 4270 nM T25258 CN35MZ 4970131 IC50 = 14500 nM T25258 C8PN0C 5280682 IC50 = 13000 nM T25258 CD64CJ 5319259 IC50 = 16000 nM T25258 CQ9GX3 5320462 IC50 = 14000 nM T25258 C19DST 5320675 IC50 = 88000 nM T25258 CPHR19 5325373 EC50 > 100000 nM T25258 CJMT13 5325385 EC50 > 100000 nM T25258 C8VZ9T 5325386 EC50 > 100000 nM T25258 C81ZSW 5325387 EC50 > 100000 nM T25258 CM47KI 5351344 IC50 = 11.5 nM T25258 CTO51S 5352005 IC50 = 16000 nM T25258 CM38PJ 5376979 IC50 = 6000 ug.mL-1 T25258 C2KZF0 5476176 IC50 = 13000 nM T25258 C4P5RL 5850257 IC50 = 141253.75 nM T25258 CD73XG 6012476 IC50 = 130 nM T25258 C1HDJ5 6055715 IC50 = 20720 nM T25258 CFO9D1 6256073 IC50 > 500000 nM T25258 C9AFO1 6708757 IC50 = 21 nM T25258 C9BM1L 6871267 EC50 = 159300 nM T25258 CBP60G 7647634 IC50 = 26400 nM T25258 CLIG51 9281828 IC50 = 3110 nM T25258 C3D9CO 9541180 EC50 = 300 nM T25258 CMIW83 9812710 IC50 = 100 nM T25258 C82UNW 9828532 EC50 = 900 nM T25258 C1C5GT 9846979 EC50 = 659 nM T25258 CVP2Q4 9849536 EC50 = 1770 nM T25258 CK5L6J 9904482 EC50 = 10000 nM T25258 CWPD26 9939298 IC50 = 1410 nM T25258 C6RQW1 9945282 IC50 = 20000 nM T25258 CR67GJ 9976755 EC50 = 6467 nM T25258 CEG64W 9976758 EC50 = 1500 nM T25258 CP02GZ 9978762 EC50 = 179 nM T25258 C1YC6F 9981658 EC50 = 58 nM T25258 CNZA83 9983792 EC50 = 75 nM T25258 CGC9R1 9984638 EC50 = 70 nM T25258 CKT03M 9985375 EC50 = 116 nM T25258 CQ0TZ3 10000408 EC50 = 329 nM T25258 CJU4W9 10002299 EC50 = 137 nM T25258 C7ZQ8A 10004336 EC50 = 27 nM T25258 C1BGV2 10005083 EC50 = 172 nM T25258 CWG2H3 10022009 EC50 = 3645 nM T25258 C64JVD 10027874 EC50 = 256 nM T25258 CJST80 10073584 IC50 = 6000 nM T25258 CPG5S3 10095159 EC50 = 110 nM T25258 CE6X4R 10221081 EC50 = 12000 nM T25258 C86TMI 10249395 EC50 = 377 nM T25258 CY73KI 10322450 EC50 = 942.5 nM T25258 C6Q1ZO 10347549 EC50 = 226 nM T25258 CC4EW9 10376018 IC50 > 100000 nM T25258 COI6B5 10381795 EC50 = 2322 nM T25258 C0V5QI 10394010 IC50 = 8000 nM T25258 CA1K2P 10423975 EC50 = 11520 nM T25258 CA67HZ 10424762 IC50 = 24730 nM T25258 CY31BG 10436076 EC50 = 671 nM T25258 C4NMT5 10456773 EC50 = 177 nM T25258 C19LEV 10461751 Ki = 630 nM T25258 C4WK3R 10471455 EC50 = 1059 nM T25258 C0DAZ6 10497861 EC50 = 8380 nM T25258 CGJ4H9 10500327 EC50 = 1741 nM T25258 CMQ29K 10503028 EC50 = 12590 nM T25258 CE1U9A 10517005 EC50 = 49700 nM T25258 CHY15F 10524623 EC50 = 83180 nM T25258 C3AYI5 10526890 EC50 = 1060 nM T25258 CXCS24 10548953 EC50 = 72440 nM T25258 C3DZM7 10550864 EC50 = 7760 nM T25258 CP5X4J 10573453 EC50 = 81280 nM T25258 CM2I4H 10577412 IC50 = 50 nM T25258 CQHL97 10589674 EC50 = 14310 nM T25258 C7U5JX 10591726 EC50 = 11030 nM T25258 CE4O3V 10596143 EC50 = 915 nM T25258 CA9YT2 10598909 EC50 = 465 nM T25258 C2R6VL 10598951 EC50 = 147 nM T25258 CU50FH 10619362 EC50 = 1210 nM T25258 C3MOA5 10620592 EC50 = 28210 nM T25258 CIE5C9 10643820 EC50 = 1807 nM T25258 C9TY3Q 10644631 EC50 = 1036 nM T25258 CI2S6D 10667675 EC50 = 299 nM T25258 CF3B5T 10692320 EC50 = 658 nM T25258 CIOL78 10699195 IC50 = 1400 nM T25258 CB51ZL 10738043 EC50 = 10070 nM T25258 CF1UM5 10746774 IC50 = 8000 nM T25258 C1CTI8 10791828 EC50 = 890 nM T25258 CUQ9Y1 10809377 EC50 = 24120 nM T25258 CA2Z9O 10809752 EC50 = 242 nM T25258 C9HD1W 10811691 EC50 = 72440 nM T25258 C75IUG 10812799 EC50 = 2690 nM T25258 CS7YZ0 10827573 EC50 = 67000 nM T25258 C18UVB 10832891 EC50 = 6875 nM T25258 CLC02T 10834768 EC50 = 123030 nM T25258 CG7YO4 10836448 EC50 = 307 nM T25258 C38GIB 10887010 Ki = 7720 nM T25258 CFC7P2 10897232 IC50 = 1550 nM T25258 CADE01 10941522 Ki = 707.95 nM T25258 CO61VZ 11161166 IC50 = 68000 nM T25258 C8P0AO 11176112 EC50 = 1550 nM T25258 C4GX9Z 11191616 Ki = 6918.31 nM T25258 C3FL9M 11199480 IC50 > 100000 nM T25258 CIQG12 11203290 Ki = 9772.37 nM T25258 CZY2I0 11225024 EC50 = 1120 nM T25258 CL1YX5 11246927 IC50 = 7330 nM T25258 C63OKC 11267785 IC50 = 1200 nM T25258 CO5UN3 11304687 EC50 = 730 nM T25258 C59RDY 11314650 EC50 = 537 nM T25258 CH4Z9E 11318780 Ki = 18197.01 nM T25258 CV68RO 11353531 Ki = 8460 nM T25258 CU5KQ1 11363211 EC50 = 2535 nM T25258 C4RLW0 11368874 IC50 > 100000 nM T25258 CEYZ65 11372107 EC50 = 3475 nM T25258 C8BM4N 11385596 EC50 = 74 nM T25258 CV3KI2 11405998 EC50 = 249 nM T25258 CB1X0H 11410427 Ki = 4250 nM T25258 CN8S6B 11417286 EC50 = 972 nM T25258 CYT3H9 11428594 EC50 = 424 nM T25258 CI97ST 11444678 Ki = 2511.89 nM T25258 C5ZYN3 11445402 Ki = 1698.24 nM T25258 C6IX1Y 11456216 Ki = 2691.53 nM T25258 C1Y4PL 11534126 IC50 < 1000 nM T25258 C57TKI 11565665 IC50 = 42000 nM T25258 C7IDH9 11596524 IC50 = 7500 nM T25258 CLJ81E 11630507 IC50 = 23000 nM T25258 C6SGF3 11644985 IC50 = 73000 nM T25258 CJK78Z 11652152 IC50 = 34000 nM T25258 CH3S9K 11666294 IC50 = 58000 nM T25258 C95EPO 11666668 IC50 = 23000 nM T25258 CJ89UZ 11687939 IC50 > 100000 nM T25258 C7RDH3 11709536 IC50 > 100000 nM T25258 CW9L4T 11723974 EC50 = 2479 nM T25258 CY8X3L 11725758 EC50 = 416 nM T25258 C7XW2Y 11742698 EC50 = 172 nM T25258 CE34NU 11757016 EC50 = 210 nM T25258 CS8DP3 11763676 Ki = 1621.81 nM T25258 C5RUT2 11787645 IC50 = 176.1 nM T25258 C4KRM1 11793594 EC50 = 9540 nM T25258 C58OBH 11794374 EC50 = 1727 nM T25258 CFV41G 11794905 EC50 = 203 nM T25258 CW73AL 11796456 EC50 = 11750 nM T25258 C07ILY 11799357 EC50 = 717 nM T25258 CGHO31 11800669 EC50 = 723 nM T25258 CZN29J 11813472 IC50 = 6100 nM T25258 CZ0H9P 11841636 IC50 = 650 nM T25258 CXLW54 11948707 Ki > 10000 nM T25258 C2C3WI 11957988 IC50 = 331.13 nM T25258 C8IFT7 11973922 EC50 = 17200 nM T25258 C9IH7R 11973925 EC50 = 27600 nM T25258 CS7U5H 11973926 EC50 > 1000000 nM T25258 CSFD67 11995339 EC50 = 95600 nM T25258 CG1CU7 12219475 EC50 > 100000 nM T25258 CS4D6C 12405466 EC50 = 3000 nM T25258 C4D7RX 12613559 EC50 = 46000 nM T25258 CH1O8Z 13113660 IC50 = 27.12 nM T25258 C6UJA5 13144102 EC50 > 100000 nM T25258 CQ3VK5 13374981 EC50 = 901 nM T25258 CV09UY 13504844 EC50 = 341 nM T25258 CH4KA7 13565926 EC50 = 230 nM T25258 C8UFO5 13984204 IC50 = 49 nM T25258 C0Q5SL 14033977 IC50 = 20640 nM T25258 CF5R6I 14057200 IC50 = 135.9 nM T25258 C4C8GW 14133592 IC50 = 15000 nM T25258 CWTY83 14338814 EC50 = 1920 nM T25258 CS5W8O 14414924 Ki = 2344.23 nM T25258 C5X3KT 14626533 IC50 = 45700 nM T25258 CD0R5N 14821386 EC50 > 100000 nM T25258 CQ89FS 14821388 EC50 > 100000 nM T25258 CNZK34 14976661 EC50 = 23180 nM T25258 CJ9Z4M 15290116 EC50 = 55400 nM T25258 CH2EY3 15837898 EC50 = 212 nM T25258 CH06TZ 15837899 EC50 = 142 nM T25258 C0RN6B 15841042 IC50 = 930 nM T25258 C4L3NU 15908916 EC50 = 7900 nM T25258 CS3YM0 15940304 IC50 = 2550 nM T25258 CMN38P 15944976 EC50 = 8770 nM T25258 C19FNV 15993184 IC50 = 1040 nM T25258 CLD92G 15999199 IC50 = 2450 nM T25258 CUZ29G 16062852 IC50 = 4700 nM T25258 C6Q4JE 16062854 IC50 = 2300 nM T25258 CL78EU 16108935 IC50 = 12 nM T25258 CX8R7B 16390581 IC50 = 15600 nM T25258 C05FVK 16451263 IC50 = 970 nM T25258 CMVW98 16618023 EC50 = 361 nM T25258 CW85LQ 16745311 EC50 = 59 nM T25258 CR1U3B 16896487 EC50 = 357 nM T25258 CPOZ18 17375361 IC50 = 15400 nM T25258 CX06NR 17412108 IC50 = 27800 nM T25258 C8C2SE 17555821 IC50 = 59 nM T25258 COG12F 17585222 IC50 = 2810 nM T25258 C0QND4 19367952 IC50 = 58100 nM T25258 CZO5S0 19697016 IC50 = 15000 nM T25258 CP7O2V 20361784 IC50 = 9800 nM T25258 CJ4Z1L 20646908 IC50 = 9332.54 nM T25258 C59FWO 20646970 IC50 = 13489.63 nM T25258 CIZV45 20646979 IC50 = 4786.3 nM T25258 CB7T2K 20963109 IC50 = 1220 nM T25258 CJ79SK 21598495 EC50 = 1452 nM T25258 C97BIZ 21598496 EC50 = 651 nM T25258 CNX3K0 21598497 EC50 = 533 nM T25258 CA0RT5 21721874 IC50 = 107.3 nM T25258 C8Q5RE 21721877 IC50 = 44.4 nM T25258 CCJ3M5 22004538 IC50 = 8500 nM T25258 CJTU32 22217363 IC50 = 155.2 nM T25258 CFI13S 22310708 IC50 = 3490 nM T25258 C3ESV6 24178402 EC50 = 820 nM T25258 CO2I3Z 24805442 EC50 = 850 nM T25258 CKW04J 24807980 EC50 = 480 nM T25258 CJUW92 24807981 EC50 = 85 nM T25258 CPO45A 24807982 EC50 = 900 nM T25258 C2VI8L 24807985 EC50 = 12000 nM T25258 C6IO1A 24807986 EC50 = 5200 nM T25258 CP8H2D 24807987 EC50 = 750 nM T25258 CAN0W4 24808151 EC50 = 1600 nM T25258 C6WUQ9 24808152 EC50 = 18000 nM T25258 C2JC1W 24808153 EC50 = 20000 nM T25258 C1HU5F 24808154 EC50 = 3100 nM T25258 C9T7BZ 24808155 EC50 = 800 nM T25258 C9SMO0 24808156 EC50 = 250 nM T25258 CW4EM8 24808157 EC50 = 650 nM T25258 CQ9LK5 24808342 EC50 = 2500 nM T25258 C7UV4H 24808344 EC50 = 180 nM T25258 C39SHG 24882446 IC50 = 144.54 nM T25258 CHB0O8 24945014 EC50 = 4860 nM T25258 C68KLJ 24945105 EC50 = 15000 nM T25258 CCS6Y4 24945108 EC50 = 35500 nM T25258 CRSQ32 24945109 EC50 = 83700 nM T25258 CAD8W3 24945110 EC50 = 31600 nM T25258 C03EIS 24945194 EC50 = 8150 nM T25258 CS9NF7 24945195 EC50 = 10200 nM T25258 C9IJX6 24945196 EC50 = 17900 nM T25258 CMU32H 25016917 Ki = 280 nM T25258 C86ZAF 25016918 Ki = 290 nM T25258 C60EJI 25113688 EC50 = 690 nM T25258 C5CGI0 25149235 Ki = 770 nM T25258 CQT4X5 25149236 Ki = 420 nM T25258 C7U6EW 25149422 Ki = 1040 nM T25258 CW2PL7 25155850 IC50 = 2500 nM T25258 C4UXF6 25155851 IC50 = 2650 nM T25258 C65LWZ 25156129 IC50 = 6500 nM T25258 CS3Q4N 25156130 IC50 = 25000 nM T25258 CZ04VO 25156131 IC50 = 14000 nM T25258 C6MXE3 25156132 IC50 = 1270 nM T25258 CU5C7V 25156133 IC50 = 5300 nM T25258 C65FNY 25156411 IC50 = 2120 nM T25258 CKIH98 25156412 IC50 = 2000 nM T25258 C35NHX 25156413 IC50 = 200 nM T25258 C94OIG 25156414 IC50 = 2500 nM T25258 C1IEF6 25156415 IC50 = 6820 nM T25258 CL1B2G 25156416 IC50 = 500 nM T25258 CUX0F4 25156684 IC50 = 80 nM T25258 CB4A2S 25156685 IC50 = 750 nM T25258 CJO48V 25156686 IC50 = 190 nM T25258 CF27EQ 25156688 IC50 = 3200 nM T25258 C8U6PV 25156966 IC50 = 1790 nM T25258 C05TOB 25157253 IC50 = 1200 nM T25258 CYM3H9 25157257 IC50 = 1200 nM T25258 CS0E3J 25157260 IC50 = 800 nM T25258 CQI4S2 25157543 IC50 = 150 nM T25258 C6Y4AJ 25157546 IC50 = 12000 nM T25258 CKP10W 25157549 IC50 = 3170 nM T25258 C9B0UR 25157845 IC50 = 140 nM T25258 CX2CP8 25157848 IC50 = 110 nM T25258 C1XP3Q 25157850 IC50 = 1720 nM T25258 C5J4ES 25158433 IC50 = 1800 nM T25258 COK46A 25158434 IC50 = 40000 nM T25258 CQRL83 25158435 IC50 = 5800 nM T25258 C26IMW 25158436 IC50 = 10000 nM T25258 C2YA4G 25217469 IC50 = 9550 nM T25258 CM80XH 25222999 IC50 > 29000 nM T25258 CSRV83 25223000 IC50 > 10000 nM T25258 C26ZQR 25223001 IC50 > 20000 nM T25258 C0S7AF 25223002 IC50 > 6000 nM T25258 CZ4A5K 25223105 IC50 > 17000 nM T25258 CKY89F 25223106 IC50 > 15000 nM T25258 CIJU21 25223199 IC50 = 9450 nM T25258 CUZ5S9 25223200 IC50 > 34000 nM T25258 C03FQV 25223201 IC50 > 57000 nM T25258 C8S6UH 25223298 IC50 > 14000 nM T25258 CZQE36 25223299 IC50 > 15000 nM T25258 C6O2ZR 25225119 EC50 = 1940 nM T25258 CM47UV 25233117 IC50 = 34.4 nM T25258 C3J8PO 39176758 IC50 = 1400 nM T25258 CI4AK1 39969954 IC50 = 31000 nM T25258 CE2RN1 42636939 IC50 = 220 nM T25258 CO9M8H 42647274 IC50 = 2100 nM T25258 C80DPH 44139216 IC50 = 5300 nM T25258 CJD3V9 44139218 IC50 = 14000 nM T25258 C6X4HN 44139220 IC50 = 14000 nM T25258 C1I2UD 44139344 IC50 > 100000 nM T25258 CB16RO 44139346 IC50 = 7900 nM T25258 C9KV0P 44139461 IC50 = 20000 nM T25258 C9VQY2 44139463 IC50 = 9000 nM T25258 CN9AH3 44139465 IC50 = 5300 nM T25258 C9BNA1 44248179 EC50 = 264 nM T25258 C4DBF9 44257640 IC50 = 19000 nM T25258 COC9A5 44265030 IC50 = 6200 nM T25258 C1R2QU 44285474 IC50 = 15000 nM T25258 C2I6MQ 44285570 IC50 = 5900 nM T25258 CU92DC 44285571 IC50 = 18100 nM T25258 C9MOA2 44285572 IC50 = 42700 nM T25258 CE1UG7 44285863 IC50 = 6000 nM T25258 C20DFI 44285866 IC50 = 11700 nM T25258 CK4E6I 44285867 IC50 = 21900 nM T25258 CT3G0A 44285868 IC50 = 7500 nM T25258 CUDK29 44285881 IC50 = 6200 nM T25258 C46QSD 44285882 IC50 = 2300 nM T25258 C5SFZ9 44285895 IC50 = 5600 nM T25258 C0AJM1 44285896 IC50 = 5400 nM T25258 CGJ2E3 44285907 IC50 = 22500 nM T25258 CFP62O 44285914 IC50 = 4300 nM T25258 CBE8Y3 44285926 IC50 > 100000 nM T25258 CU8K9D 44285958 IC50 = 10400 nM T25258 C1ZYG3 44285975 IC50 = 14900 nM T25258 CY13QV 44286211 IC50 = 16000 nM T25258 CPS2I8 44286222 IC50 = 42200 nM T25258 CS0LP4 44286259 IC50 = 17100 nM T25258 C7ZYM4 44299404 IC50 > 50000 nM T25258 C8MJP9 44364293 EC50 = 678 nM T25258 CY95IQ 44364330 EC50 = 173 nM T25258 CM0W7X 44364347 EC50 = 1536 nM T25258 CS12ZE 44364434 EC50 = 610 nM T25258 CX2SE3 44364497 EC50 = 797 nM T25258 CYI6B8 44382066 EC50 = 3700 nM T25258 C16JWF 44382121 EC50 > 10000 nM T25258 CL46DK 44382181 EC50 = 4100 nM T25258 CSP8M7 44382279 EC50 = 2300 nM T25258 C5PV0G 44382380 EC50 > 10000 nM T25258 C1NXL6 44382383 EC50 = 1130 nM T25258 C7RXU9 44382409 EC50 > 10000 nM T25258 C8J0LX 44382410 EC50 > 10000 nM T25258 CTQJ34 44382416 EC50 = 3200 nM T25258 C63SPC 44382455 EC50 > 10000 nM T25258 CSJ8V5 44382458 EC50 = 4900 nM T25258 CIQ65B 44382493 EC50 = 4000 nM T25258 CM32ND 44382536 EC50 = 1300 nM T25258 C0WLR3 44382537 EC50 = 2100 nM T25258 CU6Q1M 44382544 EC50 >> 10000 nM T25258 CZ2GW7 44382545 EC50 >> 10000 nM T25258 CZ4A5S 44382547 EC50 = 10000 nM T25258 CD0SX1 44382548 EC50 = 640 nM T25258 CZU82N 44382595 EC50 = 1470 nM T25258 C21NQI 44382629 EC50 = 1800 nM T25258 C2Z7TF 44398590 Ki = 5740 nM T25258 C4R8EB 44410932 IC50 > 100000 nM T25258 CV5H7A 44411699 IC50 = 5720 nM T25258 CSB8I1 44411703 IC50 = 4230 nM T25258 C2YGR9 44420789 EC50 > 250000 nM T25258 CG5L9N 44420793 EC50 = 820 nM T25258 C8U4PY 44420815 EC50 = 6 nM T25258 C4CVI9 44420823 EC50 = 13 nM T25258 CJT0W3 44421012 EC50 = 1686 nM T25258 CW4ZC3 44421013 EC50 = 396 nM T25258 CMT3X7 44421014 EC50 = 211 nM T25258 CF34BZ 44421015 EC50 = 162 nM T25258 C8GRH9 44421016 EC50 = 752 nM T25258 C4JOA0 44421017 EC50 = 125 nM T25258 CW7J4H 44421018 EC50 = 40 nM T25258 CZI15N 44421022 EC50 = 130 nM T25258 CYL9G2 44421023 EC50 = 178 nM T25258 COR49E 44421024 EC50 = 980 nM T25258 C2DRO4 44421025 EC50 = 10400 nM T25258 CG5Q4N 44421026 EC50 = 190 nM T25258 C2M3DA 44421027 EC50 = 137 nM T25258 C39LZO 44421028 EC50 = 1103 nM T25258 C1MTI3 44421029 EC50 = 210 nM T25258 CIM20J 44421030 EC50 = 145 nM T25258 C2Q7FJ 44421031 EC50 = 505 nM T25258 C4HKT8 44421032 EC50 = 259 nM T25258 CG16KE 44421033 EC50 = 17 nM T25258 C1MO2L 44421034 EC50 = 5470 nM T25258 CURB73 44421035 EC50 = 460 nM T25258 CLR1W2 44421036 EC50 = 9684 nM T25258 CGQ07Z 44421037 EC50 = 292 nM T25258 C91YZG 44421038 EC50 = 11190 nM T25258 CH7PD1 44421039 EC50 = 19 nM T25258 CW60EC 44421040 EC50 = 167 nM T25258 CNFG64 44421041 EC50 = 18 nM T25258 CIL12B 44421042 EC50 = 14 nM T25258 C3G4VJ 44421043 EC50 = 176300 nM T25258 C6REH4 44421044 EC50 = 1588000 nM T25258 CV9M7Q 44421045 EC50 = 336 nM T25258 C2AEM1 44421046 EC50 = 1349 nM T25258 CH9VG2 44421048 EC50 = 59 nM T25258 CMW9L8 44421049 EC50 = 179 nM T25258 C1K2PA 44421050 EC50 = 379 nM T25258 CBR97X 44421051 EC50 = 6658 nM T25258 CO1PI5 44421052 EC50 = 103600 nM T25258 CBO6C2 44421054 EC50 = 26 nM T25258 C8VTZ0 44421055 EC50 = 8490 nM T25258 C9C6ZA 44421056 EC50 = 1619 nM T25258 CDQ8H7 44421057 EC50 = 48920 nM T25258 CP4QT9 44421058 EC50 = 2568 nM T25258 CXMO94 44421059 EC50 = 1649 nM T25258 C1K5NB 44421060 EC50 = 200 nM T25258 CY6D1Q 44421061 EC50 = 227 nM T25258 C0D7HE 44421062 EC50 = 1006 nM T25258 CO47RI 44421063 EC50 = 192 nM T25258 C2UP8W 44421064 EC50 = 296 nM T25258 CY0D7P 44421065 EC50 = 859 nM T25258 C2RG7A 44428921 EC50 = 329 nM T25258 CGL49H 44428922 EC50 = 482 nM T25258 C2LHG1 44428923 EC50 = 648 nM T25258 CAWL05 44428924 EC50 = 124 nM T25258 CV4OI5 44429237 Ki = 2187.76 nM T25258 C2FL8U 44429238 Ki = 2884.03 nM T25258 CSY25K 44429239 Ki = 4160 nM T25258 CG4F9B 44429240 Ki = 700 nM T25258 CV0T5G 44429241 Ki = 1122.02 nM T25258 C0CV6Z 44429242 Ki = 570 nM T25258 C5A2OP 44429246 Ki = 7413.1 nM T25258 CAV13Q 44429252 Ki = 100000 nM T25258 C5DM6Y 44429255 Ki = 3450 nM T25258 C8XON9 44429258 Ki = 6606.93 nM T25258 C32EZP 44429263 Ki = 5495.41 nM T25258 CYO2B3 44429265 Ki = 4130 nM T25258 C83GSZ 44429268 Ki = 17378.01 nM T25258 CSX2R3 44429279 Ki = 100000 nM T25258 CQ78HT 44429285 Ki = 2810 nM T25258 CT7QU8 44429286 Ki = 794.33 nM T25258 C4F5VL 44429287 Ki = 1650 nM T25258 C5V9JT 44429289 Ki = 954.99 nM T25258 CYAB26 44429291 Ki = 12022.64 nM T25258 CQ6S8H 44429293 Ki = 8912.51 nM T25258 CB6WA8 44429297 Ki = 2500 nM T25258 CV2ZO8 44429308 Ki = 2920 nM T25258 C6J9YB 44429309 Ki = 1000 nM T25258 C3VMI8 44429310 Ki = 5128.61 nM T25258 CR7UE0 44429311 Ki = 4570.88 nM T25258 C1W8HN 44429312 Ki = 1040 nM T25258 CX20AZ 44429313 Ki = 1548.82 nM T25258 CQWK31 44429314 Ki = 2440 nM T25258 CHR5V9 44429315 Ki = 1500 nM T25258 CT2KC5 44429316 Ki = 1940 nM T25258 CA1Y0F 44429317 Ki = 4466.84 nM T25258 CQX86B 44429318 Ki = 3467.37 nM T25258 C3ZVG8 44429319 Ki = 575.44 nM T25258 CFH6U3 44429320 Ki = 7040 nM T25258 CDZ2I7 44429321 Ki = 1737.8 nM T25258 CLO07E 44429322 Ki = 910 nM T25258 CP3J1F 44429323 Ki = 1202.26 nM T25258 CCN4A6 44429324 Ki = 11220.18 nM T25258 C8UV9A 44429325 Ki = 1819.7 nM T25258 CD7LT0 44429326 Ki = 1220 nM T25258 CC86LX 44429327 Ki = 33850 nM T25258 C9GP2A 44429328 Ki = 1300 nM T25258 CI2Y1X 44429329 Ki = 1980 nM T25258 C34QPL 44429335 Ki = 3970 nM T25258 CP4KL5 44429337 Ki = 3010 nM T25258 C8CGF9 44429338 Ki = 1023.29 nM T25258 C6WUL9 44429339 Ki = 7585.78 nM T25258 C39NTQ 44429340 Ki = 302 nM T25258 C25AFY 44429341 Ki = 6918.31 nM T25258 CG2VN3 44429342 Ki = 7585.78 nM T25258 CNV52A 44429343 Ki = 7585.78 nM T25258 CWR06S 44429344 Ki = 2070 nM T25258 C9CPO7 44429345 Ki = 25040 nM T25258 CG8KV7 44429346 Ki = 3715.35 nM T25258 C03YNU 44429347 Ki = 1445.44 nM T25258 C5TX9Q 44429348 Ki = 1348.96 nM T25258 CR17PC 44429349 Ki = 724.44 nM T25258 C6SR9V 44429350 Ki = 1258.93 nM T25258 CZS1T7 44438016 IC50 = 812.83 nM T25258 C9EU5R 44451249 EC50 = 15200 nM T25258 CM8O3W 44451264 EC50 = 6350 nM T25258 C3C5FJ 44451346 EC50 = 8200 nM T25258 C43CIH 44451513 IC50 = 4168.69 nM T25258 CMHP85 44451563 IC50 = 4073.8 nM T25258 C29SBO 44451564 IC50 = 4466.84 nM T25258 C1G2CB 44451590 IC50 = 1380.38 nM T25258 C6NW0Q 44451617 IC50 = 724.44 nM T25258 C1ENZ0 44451645 IC50 = 3162.28 nM T25258 CB0OL9 44451671 IC50 = 776.25 nM T25258 CC9LK5 44451719 IC50 = 208.93 nM T25258 CS4RX9 44451745 IC50 = 630 nM T25258 C9Z4VY 44451773 IC50 = 1400 nM T25258 CTP09O 44451801 IC50 = 3162.28 nM T25258 CP69AF 44451832 IC50 = 1800 nM T25258 C45VCM 44451857 EC50 = 600 nM T25258 C4T5UP 44451866 IC50 = 3300 nM T25258 CI1Y5L 44451888 IC50 = 4897.79 nM T25258 CP3B8R 44451889 IC50 = 2238.72 nM T25258 C3S5OK 44451912 IC50 = 416.87 nM T25258 C6M3ZN 44451913 IC50 = 4168.69 nM T25258 CG61YX 44542293 EC50 > 100000 nM T25258 CI9VZ6 44542743 EC50 > 100000 nM T25258 C9AOQ4 44562411 IC50 = 1412.54 nM T25258 C4RX7I 44565362 IC50 = 850 nM T25258 CSOV56 44565422 IC50 = 2100 nM T25258 CQ1JH7 44565423 IC50 = 1400 nM T25258 CT4IY0 44565437 IC50 = 1100 nM T25258 CRS4M5 44565438 IC50 = 670 nM T25258 C6KZA1 44565439 IC50 = 1500 nM T25258 CRZ64O 44565440 IC50 = 3100 nM T25258 CR7M8S 44565458 IC50 = 3400 nM T25258 CLBO81 44565459 IC50 = 330 nM T25258 C7NRZ8 44565460 IC50 = 770 nM T25258 CW6OF8 44565479 IC50 = 670 nM T25258 CN03BJ 44565480 IC50 = 1500 nM T25258 C38FXL 44565481 IC50 = 21000 nM T25258 CZUI80 44565482 IC50 = 19000 nM T25258 CW57MC 44565508 IC50 = 14000 nM T25258 CZT54M 44565509 IC50 = 31000 nM T25258 CJGX37 44566003 IC50 = 6800 nM T25258 CH8BJ7 44566025 IC50 = 23600 nM T25258 CL52JE 44576218 EC50 = 200 nM T25258 CGC19X 44590020 Ki = 510 nM T25258 CEF1O0 44590022 Ki = 1010 nM T25258 C4Q2ER 44593438 IC50 = 4100 nM T25258 C5LK3Q 44593446 IC50 = 11000 nM T25258 C51KQN 44593447 IC50 = 11000 nM T25258 C5BG9O 44612040 IC50 = 44.4 nM T25258 C80EVI 44723582 EC50 > 100000 nM T25258 CI98LN 45482801 EC50 = 1550 nM T25258 C1T6BE 45482802 EC50 = 560 nM T25258 C5IL1C 45482820 EC50 = 3980 nM T25258 CPN3Q9 45482824 EC50 = 1100 nM T25258 CI5AT7 45482838 EC50 = 1210 nM T25258 CO46CJ 45482850 EC50 = 2250 nM T25258 C2G6BM 45482851 EC50 = 1520 nM T25258 CP0D5O 46225840 EC50 = 6290 nM T25258 C6ICB7 46225841 EC50 = 3300 nM T25258 C1P8IG 46225842 EC50 = 2230 nM T25258 C27FBP 46225896 EC50 = 390 nM T25258 C2FSL7 46225905 EC50 = 240 nM T25258 CUR03H 46225906 EC50 = 360 nM T25258 C5IS8G 46225907 EC50 = 60 nM T25258 C5O6BP 46225908 EC50 = 480 nM T25258 C3G1VI 46225925 EC50 = 5120 nM T25258 C34YIQ 46225936 EC50 = 15520 nM T25258 C8NOK5 46225937 EC50 = 890 nM T25258 C28QBM 46225938 EC50 = 40 nM T25258 C5SVN1 46225939 EC50 = 230 nM T25258 CU15AT 46225940 EC50 = 40 nM T25258 C0U6AP 46225941 EC50 = 4970 nM T25258 CRHG31 46225948 EC50 = 460 nM T25258 CUBS96 46505770 IC50 = 3548.13 nM T25258 CX2EU1 46843551 EC50 = 52600 nM T25258 CON7Q5 46888534 EC50 = 2230 nM T25258 C53NLD 46888535 EC50 = 2260 nM T25258 CWO79T 46899560 EC50 = 3350 nM T25258 CUFI19 46899561 EC50 = 4600 nM T25258 C43WPR 46899562 EC50 = 3310 nM T25258 C2QX3P 46899563 EC50 = 2150 nM T25258 CBWT20 46899565 EC50 = 20500 nM T25258 CHR49C 46899724 EC50 = 32200 nM T25258 CZXN91 46899725 EC50 = 50000 nM T25258 C7ZS6E 46899726 EC50 = 7400 nM T25258 CA3P0O 46938744 IC50 = 1680 nM T25258 CGR27B 46938838 IC50 = 730 nM T25258 CO2KM0 46938839 IC50 = 1130 nM T25258 CJA08U 46938840 IC50 = 220 nM T25258 CY4XL9 50806112 IC50 = 13400 nM T25258 C1SA2Z 53249089 IC50 = 20000 nM T25258 CG8F0J 53316757 IC50 = 20 nM T25258 CZ85PR 53317176 IC50 = 7200 nM T25258 CL8KX3 53319398 IC50 = 350 nM T25258 CHB6X4 53325051 IC50 = 24000 nM T25258 C8J5OM 53361487 Ki > 2230 nM T25258 C5CTA9 53376061 Ki > 2230 nM T25258 CWG01C 53376062 Ki > 2230 nM T25258 CU06ZF 53376063 Ki = 1340 nM T25258 C1D3IV 53376064 Ki > 2230 nM T25258 CYD8I0 53376281 Ki > 2230 nM T25258 CQBP56 53376587 Ki = 480 nM T25258 CAS3Z4 53376588 Ki = 940 nM T25258 CSEC41 53376589 Ki > 2230 nM T25258 CF7OJ2 53376698 Ki > 2230 nM T25258 C68IQN 53376699 Ki = 1780 nM T25258 CK2NS6 53376700 Ki > 2230 nM T25258 C0LFI4 53376807 Ki = 1010 nM T25258 C0RGU4 53376809 Ki = 730 nM T25258 C7D4FJ 53376810 Ki = 320 nM T25258 C2F3HN 53376811 Ki = 120 nM T25258 C3WBF4 53376918 Ki = 470 nM T25258 CJ26ZI 53376919 Ki = 220 nM T25258 C0JIZ8 53376922 Ki = 1710 nM T25258 C4Z7MF 54580539 IC50 > 1000 nM T25258 C96NWY 54580541 IC50 > 100000 nM T25258 CN30LW 54581539 IC50 > 50000 nM T25258 C6AIG3 54582535 IC50 > 50000 nM T25258 CY24RJ 54582627 IC50 > 50000 nM T25258 CN38OK 54583506 IC50 > 50000 nM T25258 CLTM38 54586400 IC50 > 50000 nM T25258 CK52PH 54586413 IC50 > 50000 nM T25258 CIAU38 54587418 IC50 > 100000 nM T25258 CKZ01T 54587433 IC50 > 100000 nM T25258 CA3C5R 54753269 EC50 = 460 nM T25258 C5UW8N 56589608 Ki = 380 nM T25258 CPY0I1 56589618 Ki = 390 nM T25258 C5A9HZ 56640837 Ki = 640 nM T25258 C8DUF3 56640861 EC50 = 6090 nM T25258 C6KDC7 56640967 Ki = 570 nM T25258 C3Y7FU 56642787 Ki = 340 nM T25258 CEQ4D2 56642788 Ki = 590 nM T25258 CDLS91 56642790 Ki = 470 nM T25258 C5TKQ4 56649310 IC50 = 1380.38 nM T25258 CM6K4Z 56658381 IC50 = 890 nM T25258 CQN29P 56658382 IC50 = 2270 nM T25258 CQ28RJ 56661871 IC50 = 4790 nM T25258 C4WQR9 56661874 IC50 > 2730 nM T25258 C4ZXU0 56663543 Ki > 2230 nM T25258 CE75GW 56665339 IC50 = 2730 nM T25258 C3PC9Q 56665340 IC50 = 2110 nM T25258 CX1EK7 56666729 Ki = 1710 nM T25258 CHP8I7 56666992 Ki = 320 nM T25258 CNRG87 56668768 IC50 = 390 nM T25258 C9U4OG 56668769 IC50 = 7420 nM T25258 CY7Z8L 56670474 Ki = 510 nM T25258 C1V2CB 56672239 IC50 > 31000 nM T25258 CG2X0M 56672240 IC50 = 360 nM T25258 CS7YT9 56672241 IC50 = 1100 nM T25258 C0EM7K 56673920 Ki > 2230 nM T25258 CLHU01 56675643 IC50 = 180 nM T25258 CF8U7D 56675645 IC50 = 1660 nM T25258 CXBM90 56678957 IC50 > 2700 nM T25258 CBH9T3 56682278 IC50 = 5770 nM T25258 C5GM4K 56682279 IC50 > 8960 nM T25258 C1H9ML 56764960 IC50 = 4830 nM T25258 C2WYN9 56945196 IC50 = 600 nM T25258 C7RW8P 56945197 IC50 > 1000 nM T25258 C7LDX6 56945198 IC50 = 400 nM T25258 C2N8DS 56945199 IC50 = 34000 nM T25258 CN2WF6 56945201 IC50 = 1300 nM T25258 CB7W4E 56945202 IC50 = 6600 nM T25258 CT4BW6 56945299 IC50 > 100000 nM T25258 CTEJ21 56945300 IC50 > 100000 nM T25258 CU2HC7 56945301 IC50 = 39100 nM T25258 CUK5Q9 56945302 IC50 = 40300 nM T25258 C36HTV 56945303 IC50 = 72000 nM T25258 C7X2EU 56945304 IC50 = 38400 nM T25258 C4VNX9 56945305 IC50 = 65000 nM T25258 C1JCB9 56945418 IC50 = 40200 nM T25258 C6UD7F 56945419 IC50 = 31200 nM T25258 C98UJH 56945420 IC50 = 67000 nM T25258 C51PRX 56945421 IC50 = 16800 nM T25258 CES25H 56945422 IC50 > 100000 nM T25258 C2QB4L 56945423 IC50 = 9100 nM T25258 CA6UX7 56945524 IC50 = 3100 nM T25258 C4AVC1 56945525 IC50 = 32500 nM T25258 CC25LY 56945526 IC50 > 100000 nM T25258 C8KLW6 56945527 IC50 > 100000 nM T25258 C6ZSA3 56945528 IC50 = 14100 nM T25258 C2IAL8 56945529 IC50 > 100000 nM T25258 CP6G0O 56945530 IC50 = 3500 nM T25258 C27RQI 56946614 IC50 = 1500 nM T25258 CK1ZU5 56946616 IC50 = 72000 nM T25258 C73GCK 56946617 IC50 > 100000 nM T25258 CL8Z0F 56946723 IC50 > 100000 nM T25258 CIQ64Z 56946724 IC50 = 31700 nM T25258 CXMK07 56946726 IC50 = 7200 nM T25258 CRY4C6 56946727 IC50 > 100000 nM T25258 CV29FO 56946728 IC50 = 1900 nM T25258 CI69QT 56946831 IC50 = 570 nM T25258 CDPU29 56946832 IC50 = 17300 nM T25258 C69ELZ 56946833 IC50 = 6800 nM T25258 CH7M4O 56946835 IC50 = 200 nM T25258 CP1VK5 56951135 IC50 = 15800 nM T25258 CU5BD9 57336812 EC50 = 202 nM T25258 CE26DW 57384779 IC50 = 80 nM T25258 C50LDI 57384780 IC50 = 170 nM T25258 CZ7UI5 57385022 IC50 = 580 nM T25258 C5XZ4I 57385023 IC50 = 3550 nM T25258 CD1XY5 57385024 IC50 = 13370 nM T25258 C1C9DI 57385271 IC50 = 200 nM T25258 CP2TG5 57385272 IC50 = 480 nM T25258 CEWB26 57385273 IC50 = 380 nM T25258 C4CDI3 57385274 IC50 = 50 nM T25258 CGR3X7 57385523 IC50 = 9480 nM T25258 C1XCE9 57393400 IC50 > 100000 nM T25258 C76TYD 57393522 IC50 = 18000 nM T25258 C7SC4L 57523668 IC50 = 111000 nM T25258 CW7B0M 57614266 IC50 = 12000 nM T25258 C8Q9ST 59051184 IC50 = 1210 nM T25258 CGRY19 70295239 IC50 = 15200 nM T25258 CXP2M4 70428348 IC50 = 48200 nM T25258 CUF6W9 70677541 IC50 = 15000 nM T25258 CIW7X5 70677689 IC50 = 17000 nM T25258 CYAO67 70681886 IC50 = 2800 nM T25258 C7Y5US 70684006 IC50 = 4500 nM T25258 CKZ3X2 70688272 IC50 = 3600 nM T25258 CWID72 70688273 IC50 = 2900 nM T25258 CY6B1N 70690284 IC50 = 6200 nM T25258 CU7F4X 70690285 IC50 = 2700 nM T25258 CV1JC6 70691873 IC50 = 15500 nM T25258 CIL5P8 70694496 IC50 = 4600 nM T25258 C6ZM8J 70696553 IC50 = 6100 nM T25258 CA1WO9 70696907 IC50 = 9300 nM T25258 CJXP74 71061793 EC50 = 1000 nM T25258 CA2N0L 71062020 EC50 = 5200 nM T25258 C0QGU2 71062093 EC50 = 2300 nM T25258 CE1QO3 71296003 IC50 = 5430 nM T25258 C93RKG 71450544 IC50 = 56000 nM T25258 CTG6I2 71450546 IC50 = 7100 nM T25258 CX52RZ 71454161 IC50 = 8700 nM T25258 CY65TU 71454163 IC50 = 9300 nM T25258 C5T0NL 71454923 IC50 = 1860 nM T25258 CTL32M 71455892 IC50 = 9600 nM T25258 C1MG4K 71459600 IC50 = 14000 nM T25258 CW97HM 71459602 IC50 > 100000 nM T25258 CAW2B8 71461339 IC50 = 10000 nM T25258 CP26MV 71461341 IC50 = 1100 nM T25258 C0FWV8 71462482 Ki = 280 nM T25258 C8RQ6M 71468723 Ki = 1010 nM T25258 COI82Z 71492427 IC50 = 147.7 nM T25258 CKMF95 71492428 IC50 = 19.5 nM T25258 C6PHS7 71492429 IC50 = 112.9 nM T25258 CT30MS 71492430 IC50 = 12 nM T25258 C3EW0F 71492431 IC50 = 97.1 nM T25258 CTC45Y 71492587 IC50 = 53.3 nM T25258 CSY29W 71492588 IC50 = 36 nM T25258 C2ZC5Q 71492589 IC50 = 14.8 nM T25258 C4ZD2W 71492590 EC50 = 214 nM T25258 C0P6IG 71492759 IC50 = 3 nM T25258 CH3M6V 71492763 IC50 = 32.2 nM T25258 CNW16J 71494857 IC50 = 45.2 nM T25258 CY82SI 71508228 IC50 = 20 nM T25258 CAQ08E 71508287 IC50 = 50 nM T25258 CV9QS7 71524587 EC50 = 2900 nM T25258 C7JIG6 71524588 EC50 = 1800 nM T25258 C1EY6B 71524589 EC50 = 600 nM T25258 C4LPZ3 71524590 EC50 = 3500 nM T25258 C60ZQJ 71524591 EC50 = 4800 nM T25258 CZ3NR9 71524817 IC50 = 72 nM T25258 C21NDB 71524818 IC50 = 29.1 nM T25258 CGV8F5 71525288 EC50 = 7100 nM T25258 CO9ZJ3 71560809 EC50 = 19000 nM T25258 C0E6OM 71560810 EC50 = 11000 nM T25258 C3T8ZF 71560811 EC50 = 250 nM T25258 CFN89Y 71560812 EC50 = 950 nM T25258 C42SMF 71560938 EC50 = 510 nM T25258 C98LPJ 71560939 EC50 = 410 nM T25258 CG8DU1 71618156 EC50 = 3700 nM T25258 C9RD7L 71624435 IC50 = 5420 nM T25258 CGA8B3 71624544 IC50 = 5990 nM T25258 CI7QT2 71624546 IC50 = 4490 nM T25258 CA7P8Q 71624648 IC50 = 10900 nM T25258 CMA90D 71624650 IC50 = 18000 nM T25258 C3KVP8 71624651 IC50 = 1230 nM T25258 CN6Q3L 71696716 EC50 = 201 nM T25258 CZ73EI 71716167 IC50 = 80 nM T25258 CT0WU5 71716785 IC50 = 75 nM T25258 C8HJM3 71717292 IC50 = 5800 nM T25258 CU4W7M 71722580 EC50 = 1367 nM T25258 C7ZR1Q 71722875 EC50 = 1310 nM T25258 CQCF98 71724480 EC50 = 300 nM T25258 C1PR7Z 71724504 EC50 = 155 nM T25258 CA7K8Z 71724506 EC50 = 746.7 nM T25258 CD9KH7 71724532 EC50 = 155.7 nM T25258 CWR2L5 71724556 EC50 = 420 nM T25258 C4ODQ2 71724557 EC50 > 1000 nM T25258 C7T0UM 71724558 EC50 = 605 nM T25258 CUL9E2 71724582 EC50 = 678.8 nM T25258 CNW68B 71724606 EC50 > 1000 nM T25258 CCZ9B3 71724628 EC50 = 360 nM T25258 C21YZQ 72722778 EC50 = 210 nM T25258 C48CAR 72735227 IC50 = 11760 nM T25258 CXWG13 72735229 IC50 = 9560 nM T25258 CFL45O 72735407 IC50 = 18210 nM T25258 C8KE4O 72737217 EC50 = 93.5 nM T25258 C9J3AP 72737219 EC50 = 110 nM T25258 C9V4FA 72793813 IC50 = 1500 nM T25258 C6NK0L 72793833 IC50 = 1500 nM T25258 C8KYL0 72793835 IC50 = 2000 nM T25258 CQ5NB6 72950792 IC50 = 21900 nM T25258 CMV14A 73293918 IC50 = 16.4 nM T25258 CO2FG6 73345390 IC50 > 2910 nM T25258 C5F4AU 73345391 IC50 = 2150 nM T25258 CKIS09 73345687 IC50 > 30000 nM T25258 C8E4UR 73345688 IC50 = 5700 nM T25258 CQV3B1 73346914 IC50 = 2680 nM T25258 C29SZY 73347040 IC50 = 17000 nM T25258 C53FHD 73347181 IC50 = 8400 nM T25258 C1MSA3 73347182 IC50 = 2000 nM T25258 C5GZR7 73347183 IC50 = 50000 nM T25258 C2GP9J 73347184 IC50 = 8100 nM T25258 CYAM67 73347185 IC50 = 2200 nM T25258 C8XU3O 73347186 IC50 = 1500 nM T25258 CB4Z3C 73347187 IC50 = 5100 nM T25258 CY35VS 73347188 IC50 = 56000 nM T25258 C53RYT 73348696 IC50 = 13100 nM T25258 C2UMC0 73348697 IC50 > 100000 nM T25258 C8Y9BO 73348698 IC50 = 19000 nM T25258 CUV2H8 73348699 IC50 = 4300 nM T25258 C02TEP 73348700 IC50 = 15000 nM T25258 C12MUH 73348701 IC50 > 100000 nM T25258 CC26MI 73348702 IC50 = 6000 nM T25258 CS5XV4 73349997 IC50 = 5880 nM T25258 CZM4L3 73349998 IC50 = 1290 nM T25258 C04MXE 73350273 IC50 = 5600 nM T25258 CP76MH 73350274 IC50 = 6400 nM T25258 C9YP4V 73350275 IC50 = 130000 nM T25258 C8A0FU 73350276 IC50 = 42000 nM T25258 CS50EI 73350277 IC50 = 15800 nM T25258 C4JG5S 73350278 IC50 = 2100 nM T25258 CB0ZS5 73350279 IC50 > 30000 nM T25258 CL38VQ 73351112 EC50 = 5000 nM T25258 C2XDR1 73351500 IC50 = 7550 nM T25258 CEP90Y 73351531 IC50 = 5200 nM T25258 CVXI38 73351612 IC50 = 2300 nM T25258 CIN06P 73351778 IC50 = 7000 nM T25258 C7SBD8 73351779 IC50 > 100000 nM T25258 CNGX73 73351780 IC50 = 2000 nM T25258 C59IQV 73351781 IC50 = 14100 nM T25258 CE6H1V 73351782 IC50 > 100000 nM T25258 C18FYB 73351783 IC50 = 3400 nM T25258 CW7R6O 73351784 IC50 = 23000 nM T25258 CGK35X 73351785 IC50 = 4000 nM T25258 C6IZG9 73352966 IC50 = 1360 nM T25258 C3KW0I 73352967 IC50 = 1550 nM T25258 CYL0N2 73352968 IC50 = 1090 nM T25258 CBLS21 73352969 IC50 = 5160 nM T25258 CJBS21 73353256 IC50 = 3000 nM T25258 C17JIV 73353257 IC50 = 2700 nM T25258 C7UC3N 73353258 IC50 = 50000 nM T25258 C3WMA5 73353259 IC50 = 4000 nM T25258 C57VIN 73353260 IC50 = 1500 nM T25258 CFXP14 73353261 IC50 = 1600 nM T25258 CPNW78 73354515 IC50 = 3500 nM T25258 C4WN9O 73354611 IC50 = 2100 nM T25258 C6LP1D 73354769 IC50 = 1300 nM T25258 CXJ53K 73354770 IC50 = 8800 nM T25258 CXD51S 73354771 IC50 = 4700 nM T25258 C29SYL 73354772 IC50 = 1600 nM T25258 C0HYX7 73354773 IC50 > 100000 nM T25258 CWVT19 73354774 IC50 = 3400 nM T25258 CR1T6W 73354775 IC50 = 1900 nM T25258 CAZ13T 73356299 IC50 = 8800 nM T25258 CKN28X 73356300 IC50 > 54000 nM T25258 CGH64E 73356301 IC50 = 11100 nM T25258 CE4CK5 73356302 IC50 = 16100 nM T25258 CO4N2W 73356303 IC50 = 8000 nM T25258 CNA3X8 73356304 IC50 = 4600 nM T25258 CUVL53 73356305 IC50 = 2400 nM T25258 CQ8V6G 76316418 IC50 = 73600 nM T25258 C9T1CV 77108045 IC50 = 620 nM T25258 CS7H4R 85998614 IC50 = 44000 nM T25258 C6WH9Z 86765226 EC50 = 27 nM T25258 C75LBD 89566370 IC50 = 12000 nM T25258 C6P7NX 89566371 IC50 = 870 nM T25258 CVL3N6 89568925 IC50 = 2754.23 nM T25258 CRB93S 89784681 EC50 = 983.3 nM T25258 CG71EX 89784708 EC50 = 159.7 nM T25258 C4ZOX6 89784717 EC50 = 896.7 nM T25258 C0ZQO6 89784722 EC50 = 198.3 nM T25258 C4U5CZ 89784733 EC50 = 403.3 nM T25258 CW17YB 89784735 EC50 = 927.5 nM T25258 C0VD4P 89784742 EC50 = 365 nM T25258 CZT7B9 89784751 EC50 = 287.5 nM T25258 CH70XJ 89784752 EC50 = 383.3 nM T25258 C6MRA2 89784753 EC50 = 321 nM T25258 C1JH4L 89784756 EC50 = 966.7 nM T25258 CN1RD8 89784760 EC50 > 1000 nM T25258 C2YB6Q 89784818 EC50 = 526 nM T25258 CSK8X6 89784827 EC50 = 277.5 nM T25258 CENX80 89785043 EC50 = 370 nM T25258 CY46QV 89785047 EC50 = 264 nM T25258 CQL7T6 89785059 EC50 = 275 nM T25258 CENR59 89785064 EC50 = 960 nM T25258 CVZG56 89785117 EC50 = 630 nM T25258 CT43OU 89785127 EC50 = 141 nM T25258 C3FB6Q 89785132 EC50 = 325 nM T25258 C4S9WG 89785146 EC50 = 650 nM T25258 CCE95J 89785148 EC50 = 345 nM T25258 C9SBA1 89785178 EC50 = 773.3 nM T25258 CSI51G 89785190 EC50 = 421.7 nM T25258 CGB2P5 89785210 EC50 = 962.5 nM T25258 CTY1H5 89785238 EC50 = 285 nM T25258 CHGX10 89785254 EC50 > 1000 nM T25258 CB1FR2 89794901 EC50 > 1000 nM T25258 C43AXK 89795130 EC50 > 1000 nM T25258 C70LJV 89795278 EC50 > 1000 nM T25258 CFU4W2 89795305 EC50 > 1000 nM T25258 CVB23M 89795326 EC50 = 430 nM T25258 CX1W9Z 89795330 EC50 = 285 nM T25258 C7XG4U 89795333 EC50 = 670 nM T25258 C7W1TP 89795335 EC50 = 763.3 nM T25258 CAX9S0 89795337 EC50 > 1000 nM T25258 COB3Z9 89795340 EC50 = 313.3 nM T25258 C6BW0Q 89795341 EC50 = 210 nM T25258 COVK20 90142631 IC50 = 6300 nM T25258 CW09JH 90645056 EC50 = 212.5 nM T25258 CJ2S4R 90645057 EC50 = 210.5 nM T25258 C5OR9X 90655449 EC50 = 3100 nM T25258 C2XS5J 90655450 EC50 = 2100 nM T25258 CDZ79W 90655451 EC50 = 300 nM T25258 CD9EI5 90655452 EC50 = 3200 nM T25258 CVT62Z 90655453 EC50 = 900 nM T25258 CRT9Y6 90655454 EC50 = 7.1 nM T25258 CAP4K6 90655455 EC50 = 1300 nM T25258 C0HOI9 90655456 EC50 = 32500 nM T25258 C79ZVA 90655457 EC50 > 100000 nM T25258 C0H9TR 90655458 EC50 > 100000 nM T25258 C3O2AW 90655459 EC50 > 100000 nM T25258 CJM3F6 90655460 EC50 = 11500 nM T25258 C37HWY 90655461 EC50 = 10900 nM T25258 CUN74Z 90655462 EC50 = 43700 nM T25258 CT6QI0 90655515 IC50 = 8510 nM T25258 C4MS6D 90655516 IC50 = 645.65 nM T25258 C0DR1J 90655517 IC50 = 40 nM T25258 CU71AI 90655518 IC50 = 140 nM T25258 C60XJR 90655519 IC50 = 1737.8 nM T25258 C0E5HA 90655520 IC50 = 1148.15 nM T25258 CFZ35T 90655521 IC50 = 2630 nM T25258 CXK7Z8 90655522 IC50 = 2330 nM T25258 CV3DQ1 90655523 IC50 = 3890 nM T25258 C4SF6T 90655524 IC50 = 138.04 nM T25258 CJK68D 90655525 IC50 = 120.23 nM T25258 C3HNZ7 90655526 IC50 = 138.04 nM T25258 CZES13 90655527 IC50 = 57.54 nM T25258 C9M4JG 90655528 IC50 = 20400 nM T25258 CTZL36 90656751 IC50 = 2000 nM T25258 C9-NOV-07 90656752 IC50 = 2500 nM T25258 C63PKA 90656753 IC50 = 6500 nM T25258 C0EUD7 90656754 IC50 = 16000 nM T25258 C59HRL 90667031 IC50 = 50000 nM T25258 CAF1K7 90667032 IC50 = 10500 nM T25258 C72BJM 90667033 IC50 = 2600 nM T25258 C58FQL 90667034 IC50 = 240 nM T25258 CAYU05 90667035 IC50 = 1100 nM T25258 CJ9FH0 101134354 IC50 = 79900 nM T25258 C21ZWF 101134356 IC50 = 39900 nM T25258 C4L8XR 101685683 IC50 = 43800 nM T25258 CV15BM 101685684 IC50 = 64400 nM T25258 CHM38S 101879129 IC50 = 3420 nM T25258 C0H9DF 101891699 EC50 = 69 nM T25258 C6V5HA 101937463 IC50 = 560 nM T25258 CXHQ89 102340685 IC50 = 4340 nM T25258 CJ7VI3 102340686 IC50 = 540 nM T25258 CS1P5K 102340687 IC50 = 200 nM T25258 C93SXK 102340688 IC50 = 310 nM T25258 C86WSC 117777746 EC50 = 325 nM T25258 C9E0BT 117777811 EC50 = 436.7 nM T25258 C9YPJ7 117803128 EC50 = 560 nM T25258 C5GUV9 118708511 IC50 = 1300 nM T25258 CQLK93 118708512 IC50 = 970 nM T25258 C5F8LY 118708513 IC50 = 8210 nM T25258 CL8H6M 118708514 IC50 = 670 nM T25258 CCT4I2 118708515 IC50 = 2930 nM T25258 C7GI8W 118708516 IC50 = 8920 nM T25258 CE7Q3U 118708517 IC50 = 3300 nM T25258 C31MGA 118708518 IC50 = 5260 nM T25258 CKV6P1 118708519 IC50 = 9200 nM T25258 C1MJ4N 118708520 IC50 = 60100 nM T25258 C7WFJ3 118708521 IC50 = 3200 nM T25258 CVK89G 118708522 IC50 = 1230 nM T25258 C7G3ZV 118708523 IC50 = 67500 nM T25258 CG8S9M 118708524 IC50 = 2760 nM T25258 C9T4KE 118708525 IC50 = 18500 nM T25258 CG3LK4 118708526 IC50 = 6660 nM T25258 C42ETW 118708527 IC50 = 21600 nM T25258 CM6TL2 118715943 IC50 = 12 nM T25258 C20UMW 118715944 IC50 = 18 nM T25258 CD91KE 118715945 IC50 = 19 nM T25258 C4XB9O 118719360 EC50 = 5800 nM T25258 CN8S1A 118719361 EC50 = 910 nM T25258 CT0CU3 118719362 EC50 = 6400 nM T25258 C2ML9T 118719363 EC50 = 4300 nM T25258 CXQN27 118719364 EC50 = 8100 nM T25258 C4Z2DS 118719365 EC50 = 800 nM T25258 CIVT58 118719366 EC50 = 570 nM T25258 C60EAN 118719367 EC50 = 2000 nM T25258 CM3IC5 118719368 EC50 = 4900 nM T25258 CLUO39 118719369 EC50 = 1300 nM T25258 CS0A4K 118719370 EC50 = 930 nM T25258 CCK02O 118719371 EC50 = 1800 nM T25258 CHI20A 118719373 EC50 = 4 nM T25258 C5SEU9 118719374 EC50 = 1200 nM T25258 C3RDT1 118719375 EC50 = 230 nM T25258 CUAY30 118720769 EC50 = 7200 nM T25258 CO3JL0 118720770 EC50 = 2850 nM T25258 CKP7B4 118720771 EC50 = 1120 nM T25258 CO9T8S 118720772 EC50 = 6570 nM T25258 CAEN90 118720773 EC50 = 4490 nM T25258 C9YB2Z 118720774 EC50 = 1350 nM T25258 C9HGO6 118720775 EC50 = 2950 nM T25258 C4WF0Y 118720776 EC50 = 7660 nM T25258 CA4MU3 118720777 EC50 = 1040 nM T25258 C5YG7N 118720778 EC50 = 4580 nM T25258 CHP3Y5 118720779 EC50 = 4680 nM T25258 C7UVG3 118720780 EC50 = 1790 nM T25258 CDWP76 118720781 EC50 = 870 nM T25258 CM7LR3 118720782 EC50 = 3450 nM T25258 CA9FI1 118720783 EC50 = 1340 nM T25258 CCJS78 118720784 EC50 = 960 nM T25258 CZ09WP 118720785 EC50 = 1740 nM T25258 CX3KD0 118720786 EC50 = 700 nM T25258 CU8SA2 118722600 IC50 > 100000 nM T25258 C3M9PE 118737173 IC50 = 11000 nM T25258 CUSI65 118737177 IC50 = 32800 nM T25258 C85ZHJ 118737178 IC50 = 37200 nM T25258 CEM28H 118737180 IC50 = 7730 nM T25258 CK34FR 122177554 Ki = 780 nM T25258 CTI6K7 122177555 Ki = 420 nM T25258 CE39OS 122177557 Ki = 610 nM T25258 CS9P6K 122177558 Ki = 290 nM T25258 CI7L1R 122179372 IC50 = 34.2 nM T25258 C2SNI0 122179373 IC50 = 25 nM T25258 CS65TF 122179374 IC50 = 21.9 nM T25258 C8G7LC 122179375 EC50 = 123 nM T25258 CU6EP1 122179376 EC50 = 123 nM T25258 C67IUV 122179377 IC50 = 40.1 nM T25258 C9D1AV 122179378 IC50 = 19 nM T25258 CWR76U 122179379 IC50 = 18 nM T25258 CWV3J6 122179380 IC50 = 8.1 nM T25258 CA67IC 122179381 IC50 = 6.2 nM T25258 C76IPE 122179382 IC50 = 15.7 nM T25258 CILW38 122179383 IC50 = 13.6 nM T25258 CZO2V5 122179384 IC50 = 13.4 nM T25258 C5JR1D 122179385 IC50 = 67.1 nM T25258 C9X7WO 122179386 IC50 = 12 nM T25258 C64JUK 122179387 IC50 = 18.5 nM T25258 C40WAE 122179388 IC50 = 11.8 nM T25258 CW7X3H 122179389 IC50 = 11.6 nM T25258 CIL20J 122179390 EC50 = 147 nM T25258 C0OUW1 122179391 EC50 = 102 nM T25258 CBX2A7 122179392 EC50 = 280 nM T25258 CQN8K7 122179393 IC50 = 4.2 nM T25258 C0CET5 122179395 IC50 = 47.9 nM T25258 CW6VU5 122179396 IC50 = 36.6 nM T25258 C5KT0L 122179397 IC50 = 31.6 nM T25258 CF2JX0 122179398 IC50 = 40.7 nM T25258 C4JU1X 122179399 IC50 = 26.2 nM T25258 CA8ZR6 122179400 IC50 = 15.9 nM T25258 C6SJN8 122179401 IC50 = 9.4 nM T25258 CI24NP 122179402 IC50 = 36.5 nM T25258 CH9OU1 122179403 IC50 = 14.4 nM T25258 CQC37W 122179404 IC50 = 27.8 nM T25258 CG9RX4 122181886 IC50 = 390 nM T25258 C7TP5G 122182828 IC50 = 860 nM T25258 CUEK57 122185090 IC50 = 10.7 nM T25258 C0DI9A 122185091 IC50 = 24.6 nM T25258 CI36SB 122185092 IC50 = 13.5 nM T25258 C4PT0L 122185093 IC50 = 6.5 nM T25258 CBTL02 122185094 EC50 = 423 nM T25258 CP7BF4 122185095 IC50 = 125.8 nM T25258 C0OSX2 122185096 IC50 = 58.2 nM T25258 CYI67B 122185097 IC50 = 25.9 nM T25258 C2FA5U 122185098 IC50 = 136 nM T25258 C9H8FD 122187974 Ki > 2230 nM T25258 C03KIL 122187975 Ki = 480 nM T25258 C7ZJB1 122187976 Ki = 940 nM T25258 C2M6GI 122187977 Ki = 1780 nM T25258 C5C8SB 122187978 Ki > 2230 nM T25258 CFN7P0 122187979 Ki = 730 nM T25258 CB9HP0 122187980 Ki = 120 nM T25258 C75VXT 122187981 Ki = 470 nM T25258 CAN63R 122187982 Ki = 220 nM T25258 C6V0FS 122187983 Ki = 1340 nM T25258 C82JKI 122187984 Ki > 2230 nM T25258 C3OL7Y 122187985 Ki > 2230 nM T25258 CN5OF6 122187986 Ki > 2230 nM T25258 C7YKT0 122188030 Ki > 2230 nM T25258 CCE46L 126587406 EC50 > 1000 nM T25258 CN0LZ6 126739167 IC50 = 12900 nM T25258 C8Z2XI 127028354 IC50 = 31300 nM T25258 C8Q9DG 127028355 IC50 = 36600 nM T25258 CRI72H 127028356 IC50 > 100000 nM T25258 C5A1NO 127028392 IC50 = 3670 nM T25258 C7OUA3 127030221 Ki = 420 nM T25258 CGQ07O 127030222 Ki = 230 nM T25258 CT13WQ 127030223 Ki = 260 nM T25258 C5P8SJ 127031139 Ki = 1520 nM T25258 C5R6VX 127031140 Ki = 310 nM T25258 CB6VZ0 127031141 Ki = 540 nM T25258 CDF3H2 127031451 Ki = 500 nM T25258 CLM59E 127031452 Ki = 520 nM T25258 C7JF4U 127031453 Ki = 250 nM T25258 C7C9PV 127032979 Ki = 470 nM T25258 CZF7B4 127033279 Ki = 130 nM T25258 C72EHU 127033280 Ki = 1740 nM T25258 CVB6S4 127033289 Ki = 400 nM T25258 CN28SM 127033290 Ki = 500 nM T25258 C7LTU2 127033563 Ki = 1210 nM T25258 CM74YN 127033564 Ki = 600 nM T25258 CL8K6E 127033864 Ki = 190 nM T25258 CL8T4E 127033865 Ki = 630 nM T25258 CYJ4P5 127033866 Ki = 310 nM T25258 CF4NG0 127033867 Ki = 630 nM T25258 C6H5OU 127033868 Ki = 1340 nM T25258 CY0R2X 127034119 Ki = 320 nM T25258 CZ7F5A 127034120 Ki = 410 nM T25258 CA47RX 127034121 Ki = 240 nM T25258 CGQC47 127034130 Ki = 460 nM T25258 CM5TK4 127034131 Ki = 610 nM T25258 CHB2S5 127034390 Ki = 500 nM T25258 CUC9I4 127040367 IC50 = 83900 nM T25258 C0I9VF 127040368 IC50 = 58200 nM T25258 CJY60W 127042304 IC50 > 100000 nM T25258 CO2P8K 127042305 IC50 > 100000 nM T25258 C56HDS 127042306 IC50 > 100000 nM T25258 CRQ7U8 127042918 IC50 = 33000 nM T25258 C39PWZ 127042920 IC50 = 58500 nM T25258 C12BJD 127042944 IC50 = 32800 nM T25258 C42ZKN 127044753 IC50 = 1290 nM T25258 CA8P0B 127044754 IC50 = 8240 nM T25258 CUF52K 127044901 IC50 = 2340 nM T25258 CF3ML0 127044902 IC50 = 5570 nM T25258 CP1K0B 127044904 IC50 = 7550 nM T25258 CO3AX7 127044909 IC50 = 18800 nM T25258 C63KNP 127044910 IC50 = 32100 nM T25258 CP2U0C 127044913 IC50 = 14600 nM T25258 C9Z8XO 127045057 IC50 = 860 nM T25258 C3FG1L 127045064 IC50 = 14900 nM T25258 CO06GR 127045207 IC50 = 800 nM T25258 CM1B6D 127045208 IC50 = 420 nM T25258 CZAL20 127045209 IC50 = 7080 nM T25258 C4DH6E 127045210 IC50 = 4150 nM T25258 C6R5MV 127045214 IC50 = 480 nM T25258 CC32NP 127048633 IC50 = 12500 nM T25258 CX76MQ 127050249 IC50 = 46700 nM T25258 C10MDY 127050524 IC50 = 59.6 nM T25258 CYXN27 127051626 IC50 = 78.82 nM T25258 C4CNG5 127051628 IC50 = 73.14 nM T25258 CX20OQ 129903920 IC50 = 2080 nM T25258 CU2OD6 132574625 EC50 = 119.6 nM T25258 CN7U0O 132576652 IC50 = 8380 nM T25258 CV87LG 132576653 IC50 = 22820 nM T25258 CL98GC 132576654 IC50 = 7820 nM T25258 CV80DI 132576655 IC50 = 6930 nM T25258 C0WU3K 132576656 EC50 = 252.6 nM T25258 C06ZYL 132576657 IC50 = 4520 nM T25258 C45KEY 132576658 IC50 = 6250 nM T25258 C1V7GY 134129908 IC50 = 9400 nM T25258 CQ5N3X 134129987 IC50 = 434 nM T25258 CDG0S3 134130015 IC50 = 21800 nM T25258 C13RTP 134130119 IC50 = 4030 nM T25258 CG0NC4 134130126 IC50 = 9780 nM T25258 CA7QF6 134130525 IC50 = 3200 nM T25258 C63NSK 134130669 IC50 = 19400 nM T25258 C6LRO0 134131064 IC50 = 5470 nM T25258 CD69RC 134131216 IC50 = 2880 nM T25258 CWP09Q 134131281 IC50 = 8140 nM T25258 C1JP2L 134131336 IC50 = 10200 nM T25258 C6GIZ2 134131389 IC50 = 4200 nM T25258 CB7A2U 134131478 IC50 = 6200 nM T25258 CDJ2L0 134133476 IC50 = 16300 nM T25258 CVRT47 134134470 IC50 > 500000 nM T25258 CQO05X 134141004 IC50 > 500000 nM T25258 C3PIE7 134141342 IC50 = 12600 nM T25258 CE14NO 134156590 IC50 = 12100 nM T25258 CP5BS7 135185926 IC50 = 4 nM T25258 CL93MJ 135185931 IC50 = 192 nM T25258 CX13SP 135185932 IC50 = 7 nM T25258 CNK8Z0 135185934 IC50 = 0.78 nM T25258 CD13BT 135185936 IC50 = 11 nM T25258 CPD4H1 135185937 IC50 = 21 nM T25258 CXYD91 135185942 IC50 = 57 nM T25258 C7ZRK9 135185944 IC50 = 185 nM T25258 C6ZK3C 135449697 EC50 > 100000 nM T25258 C2WXZ5 135502061 EC50 = 3790 nM T25258 CZO0D7 135993331 EC50 = 102200 nM T25258 C1EB8Q 136236384 EC50 = 2800 nM T25258 C2EG4I 137133332 IC50 = 52720 nM T25258 CI29NG 137133333 IC50 = 17040 nM T25258 CMA71O 137133334 IC50 = 39930 nM T25258 CZF08H 137133335 IC50 = 37640 nM T25258 CH05QS 137633237 IC50 > 10000 nM T25258 CTZY18 137633964 IC50 = 5 nM T25258 C6BY4C 137634390 IC50 > 100000 nM T25258 C6S5ZA 137634903 IC50 = 3.11 nM T25258 CZ5X3J 137635158 IC50 = 85360 nM T25258 C6XEW4 137635483 IC50 = 84780 nM T25258 CI1S9R 137636359 IC50 = 2780 nM T25258 CHB5K6 137636574 IC50 = 27690 nM T25258 CW8ZJ6 137637229 IC50 = 38090 nM T25258 C8IM4P 137637833 IC50 = 3096 nM T25258 C3EB6I 137638388 IC50 = 89160 nM T25258 C42KCL 137638514 IC50 = 8730 nM T25258 C4YD3A 137639105 IC50 = 2862 nM T25258 C0T9VN 137639186 IC50 > 100000 nM T25258 C65PTM 137641138 IC50 = 17.2 nM T25258 CPXS38 137641162 IC50 = 7650 nM T25258 CE41MQ 137641298 IC50 = 510 nM T25258 CM8LO4 137643183 IC50 = 1643 nM T25258 C2HB8V 137643768 IC50 > 100000 nM T25258 C9CGU8 137644196 IC50 = 760 nM T25258 CTK3S2 137644305 IC50 = 21070 nM T25258 C67TRY 137644531 IC50 = 83860 nM T25258 CN6PY0 137645040 IC50 = 8 nM T25258 CS87DF 137645885 IC50 > 10000 nM T25258 C1VQO6 137645918 IC50 = 3231 nM T25258 C5PIW6 137646356 IC50 = 1.25 nM T25258 CJQ70A 137647200 IC50 = 26920 nM T25258 CU7E0V 137647244 IC50 = 25520 nM T25258 CZO45P 137647673 IC50 > 100000 nM T25258 CVL5T7 137648146 IC50 = 6300 nM T25258 CLV1B0 137648329 IC50 = 16740 nM T25258 C1H3PM 137648400 IC50 = 77920 nM T25258 C3G5UK 137649335 IC50 = 100 nM T25258 C18XJI 137649439 IC50 = 52300 nM T25258 CG0O8U 137649914 IC50 = 73370 nM T25258 CF0X4M 137649928 IC50 > 100000 nM T25258 CP4Q2G 137650393 IC50 = 12160 nM T25258 C3IEL0 137650562 IC50 = 14.2 nM T25258 CM9NO6 137652146 IC50 = 4.05 nM T25258 CQZC26 137652529 IC50 = 48700 nM T25258 C3JE5U 137652980 IC50 = 1296 nM T25258 CFQ2P3 137653396 IC50 = 11.22 nM T25258 CWP8Y3 137654281 IC50 > 100000 nM T25258 C3HM2S 137655403 IC50 = 21910 nM T25258 CD23EA 137655428 IC50 = 4 nM T25258 CDCB45 137655666 IC50 = 17 nM T25258 CD1L5S 137657500 IC50 = 1394 nM T25258 COXF43 137658445 IC50 = 1449 nM T25258 CFHN34 137658683 IC50 = 45210 nM T25258 C5C0KF 137658808 IC50 = 334 nM T25258 CUJ58E 137658891 IC50 > 10000 nM T25258 CAX5B2 137659144 IC50 > 100000 nM T25258 CXT19C 137660556 IC50 = 10 nM T25258 CM4U2P 137661238 IC50 = 31920 nM T25258 CEMK45 137661609 IC50 > 100000 nM T25258 C7N9HZ 137661643 IC50 = 19.9 nM T25258 CA3BV4 137661982 IC50 = 8290 nM T25258 CPI3E4 137662036 IC50 = 12700 nM T25258 CSNT57 137662263 IC50 > 100000 nM T25258 C70RHF 138454755 IC50 = 28.29 nM T25258 C5PKZ2 139593897 IC50 = 2870 nM T25258 C9USZ1 145949183 IC50 = 1100 nM T25258 CUY09I 145950988 IC50 = 1810 nM T25258 C6LNS7 145953170 IC50 = 290 nM T25258 CHCB46 145956407 IC50 = 3150 nM T25258 CO12MI 145957929 IC50 = 2.4 nM T25258 CBQ8K0 145959274 IC50 = 1670 nM T25258 C4PQ5A 145959673 IC50 = 1870 nM T25258 CYL21E 145960198 IC50 = 3260 nM T25258 C1A7DH 145964067 IC50 = 11700 nM T25258 C80ESB 145964513 IC50 = 11000 nM T25258 CM5W0B 145964551 IC50 = 5910 nM T25258 CZ4I8A 145975509 IC50 = 8550 nM T25258 CA3V5K 145976004 IC50 = 21200 nM T25258 C7HUX6 145978131 Ki = 2800 nM T25258 CF8L7A 145979103 EC50 = 489.7 nM T25258 CH0D4R 145979502 EC50 = 2000 nM T25258 C3EX7W 145979504 EC50 = 384 nM T25258 CP61TJ 145979699 EC50 = 8400 nM T25258 C9G3PT 145979902 EC50 = 6900 nM T25258 C4G7LT 145980033 EC50 = 328 nM T25258 C6TCD8 145981227 EC50 = 2540 nM T25258 C26OWY 145981942 EC50 = 333.5 nM T25258 CSHK75 145982928 EC50 = 5400 nM T25258 C13VFZ 145985646 EC50 = 68.7 nM T25258 CZIF02 145985848 EC50 = 1600 nM T25258 C4A1LN 145985882 EC50 = 1510 nM T25258 C90ZNB 145986644 EC50 = 3040 nM T25258 C30TAS 145986947 EC50 = 15200 nM T25258 CI38SJ 145987174 EC50 = 12700 nM T25258 CFU24J 145987833 EC50 = 161 nM T25258 CGL02K 145988126 EC50 = 515 nM T25258 CMH16X 145988902 EC50 = 2170 nM T25258 C2G5UB 145989426 EC50 = 11000 nM T25258 CMT4D2 145989461 EC50 = 4730 nM T25258 CX3YR7 145990226 EC50 = 349.5 nM T25258 C1EFK9 145990343 EC50 = 2800 nM T25258 CV03YM 145990388 EC50 = 6200 nM T25258 CZRB08 145990960 EC50 = 1860 nM T25258 CVSF12 145992209 EC50 = 2830 nM T25258 CN1V8K 145992500 EC50 = 255 nM T25258 CT02XU 145992768 EC50 = 218.5 nM T25258 C07OTB 145993028 EC50 = 344.4 nM T25258 C65JUT 145993130 EC50 > 1000 nM T25258 C3UC5J 145994097 EC50 = 258.8 nM T25258 CKM79V 145994277 EC50 = 88.5 nM T25258 CE9Q1N 146422024 IC50 = 6 nM T25258 C3VZL4 146430218 IC50 = 17 nM T25258 CB8J6W 154728908 IC50 = 1020 nM T25258 CF92IR 155510784 EC50 = 0.97 nM T25258 CIY5B0 155510937 IC50 = 27520 nM T25258 CXH10R 155511058 IC50 = 4900 nM T25258 CWU2Z8 155511062 IC50 = 23590 nM T25258 CYCK65 155511137 IC50 = 1590 nM T25258 CQ2S9Y 155511222 EC50 = 1100 nM T25258 C5VRT4 155511477 IC50 = 15000 nM T25258 C1L0WJ 155511549 IC50 = 380 nM T25258 CC14DU 155511650 EC50 = 1700 nM T25258 C3MZ1E 155511724 EC50 = 910 nM T25258 CE4C1X 155512695 IC50 = 660 nM T25258 CJZD76 155512908 IC50 = 90 nM T25258 CC86NH 155513586 IC50 = 7.03 nM T25258 CVZ7D2 155514151 EC50 = 810 nM T25258 C0AFT8 155514623 EC50 > 1000 nM T25258 CWKG62 155515033 IC50 = 23590 nM T25258 C17AZU 155515244 EC50 = 920 nM T25258 CU06MC 155515357 IC50 = 35.4 nM T25258 CH6O3X 155515825 EC50 = 200 nM T25258 CGPY31 155516187 EC50 = 29500 nM T25258 CV9TF6 155516191 EC50 > 1000 nM T25258 CV6OX1 155517977 IC50 = 17960 nM T25258 C4IS7E 155518051 EC50 = 220 nM T25258 CFTG31 155518068 IC50 = 20600 nM T25258 CLQO05 155518383 IC50 = 1880 nM T25258 CWNS51 155518629 EC50 = 290 nM T25258 CCK94U 155519382 IC50 = 8030 nM T25258 C6CS7Z 155519855 IC50 = 28000 nM T25258 C0DQI6 155520044 IC50 = 21780 nM T25258 CL4K9O 155520563 EC50 = 350 nM T25258 CA1BD2 155520579 EC50 = 1380 nM T25258 CXJK95 155520599 IC50 = 5000 nM T25258 C9OT7K 155521224 IC50 = 7860 nM T25258 C8WFN9 155522227 IC50 = 410 nM T25258 C8V3OE 155522345 IC50 = 190 nM T25258 CQK86M 155522385 IC50 = 330 nM T25258 CS18PU 155523410 EC50 = 710 nM T25258 CN6ST7 155523417 EC50 > 1000 nM T25258 C1V9YM 155523822 EC50 = 260 nM T25258 C71GOI 155524022 EC50 = 1520 nM T25258 C6X8DN 155524147 IC50 = 13100 nM T25258 CL61VT 155524337 IC50 = 9390 nM T25258 CP69ML 155525680 IC50 = 14200 nM T25258 CGQ31C 155525684 IC50 = 4000 nM T25258 C86ZPR 155525910 EC50 = 110 nM T25258 C8C7VA 155525927 EC50 = 0.9 nM T25258 C6YN1V 155526435 EC50 = 290 nM T25258 C8TQ4G 155526547 EC50 > 1000 nM T25258 CTW8I2 155526857 EC50 = 520 nM T25258 CJD24F 155527052 IC50 = 12900 nM T25258 C41JTR 155528166 EC50 = 930 nM T25258 C9BGT5 155528240 EC50 = 573.3 nM T25258 CCQZ80 155528271 EC50 = 21200 nM T25258 C2U1TW 155529037 IC50 = 4690 nM T25258 C75OQS 155529248 IC50 = 1420 nM T25258 CGW7P5 155529293 IC50 = 1890 nM T25258 C3O4FR 155529325 IC50 = 190 nM T25258 C56AHP 155530068 EC50 = 414.3 nM T25258 C4AE8R 155530476 IC50 = 8830 nM T25258 CVB45K 155530670 IC50 = 39950 nM T25258 C9F3YI 155530680 IC50 = 220 nM T25258 C9N3RV 155530862 IC50 = 2630 nM T25258 C1HFX4 155531129 EC50 = 1040 nM T25258 C6I0LU 155531567 IC50 = 460 nM T25258 CUL2G4 155531672 EC50 > 1000 nM T25258 C64UBA 155531687 IC50 = 13300 nM T25258 C9VWU0 155532632 IC50 = 9600 nM T25258 C4VO1R 155532870 IC50 = 12640 nM T25258 CCS6U1 155533262 IC50 = 14840 nM T25258 C6HBT0 155533347 IC50 = 17410 nM T25258 CW4L9C 155533357 IC50 = 6260 nM T25258 C4IW9M 155533366 EC50 = 310 nM T25258 C9QT4A 155533532 IC50 = 18800 nM T25258 CV2E0X 155533958 IC50 = 42310 nM T25258 C2I3DM 155533970 IC50 = 21600 nM T25258 CWT89R 155534133 EC50 = 15.3 nM T25258 CRC20Y 155534149 EC50 = 550 nM T25258 CP9C0M 155534240 IC50 = 5010 nM T25258 C1PBZ6 155534314 IC50 = 52210 nM T25258 CS9QJ1 155534558 EC50 = 1470 nM T25258 CY05LS 155534635 EC50 = 1050 nM T25258 CNUX50 155534847 EC50 = 54 nM T25258 COLA68 155535254 IC50 = 7300 nM T25258 CHF7A6 155535686 EC50 > 1000 nM T25258 CZ46CP 155536047 EC50 = 900 nM T25258 C28CPM 155536187 IC50 = 160 nM T25258 CJE5V8 155536523 IC50 = 9900 nM T25258 CQC9E5 155536529 IC50 = 280 nM T25258 COFC46 155536723 EC50 = 690 nM T25258 CGM43D 155536878 IC50 = 910 nM T25258 CP3U4C 155536912 EC50 = 320 nM T25258 C5XT8N 155536956 IC50 = 300 nM T25258 CYG84N 155537154 EC50 = 73 nM T25258 CB1FI9 155537197 IC50 = 1410 nM T25258 C2J7TM 155537461 IC50 = 1810 nM T25258 CGD47O 155537584 EC50 > 1000 nM T25258 C2MOH0 155537676 IC50 = 9500 nM T25258 CNS83Y 155538210 IC50 = 150 nM T25258 CNFV23 155538280 EC50 = 380 nM T25258 CPT8R7 155538460 IC50 = 18750 nM T25258 CVES34 155538494 EC50 = 320 nM T25258 CFN41J 155538958 EC50 = 990 nM T25258 CLU37N 155539307 EC50 = 210 nM T25258 CXN6C4 155539538 IC50 = 550 nM T25258 C1HI6G 155539765 EC50 = 6930 nM T25258 C03FHL 155541091 IC50 = 135.4 nM T25258 CS3E7W 155541094 IC50 = 59230 nM T25258 CL0WO4 155541816 IC50 = 7800 nM T25258 CE0G9A 155542384 IC50 = 8760 nM T25258 CL6QG0 155542981 IC50 = 2700 nM T25258 CP93FH 155543149 EC50 = 960 nM T25258 C7JUC3 155543680 EC50 = 300 nM T25258 C0GVI7 155545772 EC50 = 1200 nM T25258 CMIN20 155545978 IC50 = 4740 nM T25258 COB86G 155548770 EC50 = 1180 nM T25258 C68MYP 155548971 IC50 = 20070 nM T25258 CDY82R 155549328 EC50 = 760 nM T25258 C86HEA 155549333 IC50 = 22500 nM T25258 C72IFK 155549366 IC50 = 9230 nM T25258 CZ9S8E 155549957 IC50 = 3570 nM T25258 C1HI5E 155550141 IC50 = 160 nM T25258 C53PGC 155550195 EC50 = 3120 nM T25258 CWK3L0 155550287 EC50 = 910 nM T25258 CB8FC1 155550293 EC50 = 650 nM T25258 C8F3HQ 155550402 IC50 = 6550 nM T25258 C8TQB0 155550535 IC50 = 5120 nM T25258 C8B3LI 155551011 IC50 = 770 nM T25258 CGF1W0 155551433 IC50 = 6220 nM T25258 CX43TI 155551742 IC50 = 190 nM T25258 CP7A5R 155552128 EC50 = 230 nM T25258 C1ODI3 155552499 EC50 = 870 nM T25258 C0CN2Z 155552511 EC50 = 19200 nM T25258 C8LM7I 155552602 IC50 = 26560 nM T25258 CIF4T8 155553306 EC50 > 1000 nM T25258 CG9K4Y 155553476 EC50 = 1.3 nM T25258 CEZ7B1 155554618 EC50 = 480.7 nM T25258 CX6CM0 155554919 EC50 = 893.3 nM T25258 C2Y9UG 155554959 EC50 = 720 nM T25258 CU9P0W 155555392 IC50 = 1000 nM T25258 C02QZX 155555706 EC50 = 5200 nM T25258 CHYW74 155555831 IC50 = 5300 nM T25258 C7JI4C 155555932 EC50 = 204 nM T25258 C7Y0QL 155557304 IC50 = 25300 nM T25258 C7AB2T 155557729 EC50 = 3100 nM T25258 CG0H8N 155557744 EC50 = 850 nM T25258 CM2J5L 155558116 EC50 = 1400 nM T25258 CE6HB4 155558201 IC50 = 23590 nM T25258 C27XQN 155558615 EC50 = 616.3 nM T25258 C8ATZ5 155558917 IC50 = 560 nM T25258 CUNV65 155558919 EC50 = 683.2 nM T25258 C21LPY 155559292 IC50 = 23400 nM T25258 CFRS42 155559312 IC50 = 390 nM T25258 CG6NC7 155560071 EC50 = 1100 nM T25258 C46KOL 155560381 IC50 = 14300 nM T25258 CE6C4X 155562808 IC50 = 220 nM T25258 CPOI59 155562875 IC50 = 19200 nM T25258 CU9AV8 155563251 IC50 = 31600 nM T25258 CWM67C 155563340 EC50 = 550 nM T25258 CS0NC2 155563858 IC50 = 8240 nM T25258 CU1TG6 155564277 IC50 = 7400 nM T25258 C7SMU4 155565022 IC50 = 2860 nM T25258 CGV09H 155566167 IC50 = 10300 nM T25258 C6Z2XK 155566234 EC50 = 820 nM T25258 C4SNI0 155566321 IC50 = 8000 nM T25258 CG95OM 155566333 IC50 = 17960 nM T25258 CAN76P 155566986 EC50 = 0.6 nM T25258 C8ZE6S 155567126 IC50 = 11300 nM T25258 CO1LU7 155567143 EC50 > 1000 nM T25258 C2ER6P 155567163 IC50 = 16620 nM T25258 CKW4Y3 155567530 EC50 = 1200 nM T25258 C7KFG6 155567619 EC50 = 1000 nM T25258 CHT79A 155568041 EC50 = 950 nM T25258 CJ7T4M 155568050 EC50 = 21400 nM T25258 CTV5K3 155568177 EC50 > 1000 nM T25258 CTK36H 155568395 EC50 = 1170 nM T25258 C03SJY 155568508 EC50 = 245.5 nM T25258 CO08ZV 155568670 EC50 = 340 nM T25258 CN31VJ 155568802 IC50 = 410 nM T25258 CTXV81 155568869 EC50 > 1000 nM T25258 COQJ76 155569267 IC50 = 3380 nM T25258 C0K1HQ 155569340 IC50 = 70 nM T25258 CCBA65 155569529 EC50 = 3300 nM T25258 CMU7H3 155569706 EC50 = 980 nM T25258 CP9TR0 10324985 Ki > 10000 nM T25258 D00AII 5281727 IC50 = 42000 nM T25258 D03PLP 11579996 IC50 = 12000 nM T25258 D04GYT 15511439 IC50 = 251.19 nM T25258 D04TQF 11973927 EC50 = 92800 nM T25258 D05XGZ 11536458 IC50 = 16000 nM T25258 D07RSH 631105 IC50 = 27100 nM T25258 D09HIM 22004473 IC50 = 524.81 nM T25258 D09MGF 11973811 EC50 > 1000000 nM T25258 D09ROW 10212 IC50 = 28000 nM T25258 D0A4TF 15511440 IC50 = 165.96 nM T25258 D0A7AK 11973810 EC50 = 125000 nM T25258 D0AW4W 11537051 IC50 = 16000 nM T25258 D0AZ0Y 11514345 IC50 = 53000 nM T25258 D0E5IP 3795 EC50 = 3080 nM T25258 D0H4YH 11594901 IC50 = 80000 nM T25258 D0I7GE 11790 IC50 = 24600 nM T25258 D0JL2T 5393152 IC50 = 3200 ug.mL-1 T25258 D0KL1P 10474335 EC50 = 550 nM T25258 D0O9NE 5388063 IC50 = 8000 nM T25258 D0PI0R 11609210 IC50 = 28000 nM T25258 D0QG6G 11493254 IC50 = 20000 nM T25258 D0RQ8R 11973809 EC50 = 100000 nM T25258 D0S8CE 15950351 IC50 = 354.81 nM T34429 D0K0KH 656665 Ki = 6.9 nM T34429 D0LM4A 170361 Ki = 125 nM T34429 D0PG8O 5360515 IC50 = 25000 nM T34429 D0Q9HF 187 Ki = 501.19 nM T34429 D0T8GD 89594 Ki = 620 nM T34429 D0V8HA 4032 IC50 = 12300 nM T34429 D0X4ZR 444 IC50 = 50000 nM T34429 D00EZO 10176607 Ki = 6900 nM T34429 D01IVE 101616 Ki = 7943.28 nM T34429 D05LRD 59286554 Ki = 8.1 nM T34429 D08XPW 10235 Ki = 1420 nM T34429 D0D3TX 46196517 Ki = 4.3 nM T34429 D0H1AY 50914822 EC50 = 39 nM T34429 D0Y6OE 5310969 Ki = 148 nM T34429 D0ZC3C 5310985 EC50 = 1995.26 nM T34429 D03UID 5310967 Ki = 8000 nM T34429 D03YPJ 5163 EC50 = 1500 nM T34429 D04HYP 3075702 Ki = 2060 nM T34429 D09ADT 119380 Ki = 4050 nM T34429 D0AB4Q 9824145 EC50 > 10000 nM T34429 D0L1DP 178052 Ki > 10000 nM T34429 D0Q9RR 9794392 Ki = 3 nM T34429 D0Y9HH 3036156 EC50 > 10000 nM T34429 D0Z0LJ 11151363 Ki = 0.2 nM T34429 C6GO7P 412 Ki = 730 nM T34429 CJ4M1W 1316 EC50 = 31000 nM T34429 C2IUD9 2181 Ki = 450 nM T34429 C45PUM 2551 Ki = 66000 nM T34429 C9IK1Y 4136 Ki = 44000 nM T34429 C48GPY 5475 EC50 = 2500 nM T34429 C6VPU2 15548 EC50 > 100000 nM T34429 CG3D7A 22301 EC50 > 100000 nM T34429 C3VL1J 27694 EC50 > 100000 nM T34429 C8G4LA 29758 Ki = 9700 nM T34429 CGE2K7 41221 EC50 > 100000 nM T34429 C2NM4A 72503 IC50 > 100000 nM T34429 CQ8ES5 97424 Ki = 6309.57 nM T34429 CUI25G 115224 IC50 = 100000 nM T34429 CC1HD0 127922 Ki > 10000 nM T34429 CPH6Y4 155481 EC50 = 40000 nM T34429 CL3I6A 165829 IC50 = 880 nM T34429 CVP7Y4 169017 Ki = 7500 nM T34429 CP81IV 204031 Ki = 12589.25 nM T34429 C3OR0P 215992 EC50 = 10000 nM T34429 CT3Z4U 216066 Ki >= 31622.78 nM T34429 CG3BZ8 216726 Ki = 19952.62 nM T34429 CJXK79 258214 IC50 = 1150 nM T34429 CPAS21 280225 EC50 > 100000 nM T34429 CVD1E8 372331 Ki >= 31622.78 nM T34429 C2BIJ6 442343 IC50 = 3100 nM T34429 CLK6R5 521233 Ki >= 31622.78 nM T34429 CT7WN8 604334 Ki = 199.53 nM T34429 C0DBZ2 606141 IC50 = 30000 nM T34429 C3IZC4 637026 IC50 = 44000 nM T34429 C4VX6K 637578 Ki = 15848.93 nM T34429 CZ0AH3 638278 EC50 = 11600 nM T34429 C5JG9L 684225 Ki = 1949.84 nM T34429 C8QW5E 719215 Ki = 6309.57 nM T34429 CFD4A1 827143 Ki = 15848.93 nM T34429 CG0S6R 827171 Ki >= 31622.78 nM T34429 CER1D9 832487 Ki = 15848.93 nM T34429 C1T6CV 854051 Ki = 8511.38 nM T34429 C0EWM5 1067742 Ki >= 31622.78 nM T34429 CX3C0J 1761244 IC50 = 14500 nM T34429 CU4D6G 1781989 Ki >= 31622.78 nM T34429 CD4T5G 1811379 Ki >= 31622.78 nM T34429 C6AFR3 2770381 Ki >= 31622.78 nM T34429 C6D9EH 2772083 Ki = 7943.28 nM T34429 C1V5LY 2859426 Ki = 6309.57 nM T34429 CU26BM 2939361 Ki = 1995.26 nM T34429 CH81TW 3034748 Ki = 91 nM T34429 C3B1WI 3073763 EC50 = 39.81 nM T34429 CV48RU 3142092 Ki = 3981.07 nM T34429 CZ1J0H 3148804 Ki >= 31622.78 nM T34429 CK57ZE 3438145 IC50 = 30000 nM T34429 CQID37 3526851 Ki >= 31622.78 nM T34429 CP86NR 4105638 Ki = 19952.62 nM T34429 CSJ06P 4401657 Ki = 3162.28 nM T34429 C3F9PH 4658560 Ki >= 31622.78 nM T34429 CSG73K 4694339 Ki = 12 nM T34429 C7PE2V 5013705 EC50 = 10000 nM T34429 CLJ3F8 5038679 EC50 = 1300 nM T34429 CNW31R 5280960 EC50 = 4000 nM T34429 C1EVM7 5310971 Ki = 92 nM T34429 CQ3PL4 5322052 EC50 = 38000 nM T34429 CSX83Z 5333825 Ki = 5011.87 nM T34429 C7CD3G 5805298 EC50 = 1900 nM T34429 C9IF7W 5811533 EC50 = 4000 nM T34429 CM6LP8 5824382 IC50 = 110 nM T34429 CI5B1Z 5939029 EC50 = 6100 nM T34429 CBY1G2 5976625 EC50 = 17200 nM T34429 C1SP3X 5980988 EC50 = 25000 nM T34429 CMK04Z 6433339 IC50 = 41 nM T34429 CU7NH4 6474292 EC50 = 34500 nM T34429 CLY28A 6554040 EC50 = 28000 nM T34429 CJ3FS9 6603935 IC50 = 2200 nM T34429 CLM7T3 6918622 IC50 = 600 nM T34429 CUE4C9 7172378 Ki = 10232.93 nM T34429 CY1XN7 7446712 EC50 = 158.49 nM T34429 CM6X0B 7571808 EC50 = 1258.93 nM T34429 C3BH7M 8646887 EC50 = 1258.93 nM T34429 C74CBS 9794141 Ki = 1530 nM T34429 C6YDQ0 9795278 Ki = 24.55 nM T34429 CK0U5Q 9797360 Ki = 14 nM T34429 C6X3RP 9813490 Ki = 1700 nM T34429 C1M0SN 9815622 Ki = 2400 nM T34429 C71JPQ 9822806 IC50 = 8500 nM T34429 CHDY16 9834184 Ki = 350 nM T34429 C80NVH 9834302 Ki = 520 nM T34429 C5LJF4 9858016 Ki = 75 nM T34429 C0Z5RS 9859386 IC50 = 6000 nM T34429 CF72XZ 9860561 Ki = 0.03 nM T34429 COCP14 9879332 Ki = 9 nM T34429 C2C0MT 9881371 EC50 = 199 nM T34429 C7WCB6 9883332 Ki = 28 nM T34429 CRST76 9899814 Ki = 617 nM T34429 CAJ1X8 9920686 Ki = 1.6 nM T34429 CDJ34P 9921125 Ki = 25 nM T34429 CFGM25 9921468 Ki = 80 nM T34429 CA17GY 9922799 Ki = 3.4 nM T34429 C0C7NV 9930121 Ki = 7 nM T34429 COD73F 9943346 Ki = 1.6 nM T34429 C7TS9J 9944605 Ki = 16.7 nM T34429 CK4X0Y 9970311 EC50 = 100 nM T34429 CR84AX 9970357 Ki = 6 nM T34429 C9XUH5 9976826 EC50 = 5500 nM T34429 CIWG38 10015966 EC50 = 580 nM T34429 CID3J4 10019186 Ki = 167 nM T34429 C8BM4D 10044336 Ki = 112 nM T34429 CGM3W9 10059716 Ki = 7600 nM T34429 C7VX8R 10059884 EC50 = 197 nM T34429 CJD7Z9 10060963 Ki = 14454.4 nM T34429 C1N4TL 10061378 EC50 = 190 nM T34429 C7O5DA 10061682 EC50 = 4800 nM T34429 CCV98T 10107174 EC50 = 129 nM T34429 CP79CI 10130239 Ki = 420 nM T34429 CI0W5C 10130417 EC50 = 440 nM T34429 C2CT5D 10130418 Ki = 979 nM T34429 CDH4J3 10130527 IC50 = 9900 nM T34429 C6LB2N 10130752 IC50 = 4000 nM T34429 CN05GL 10176454 Ki = 40 nM T34429 CM9B2Z 10176482 Ki = 830 nM T34429 CM58IK 10219887 EC50 > 300000 nM T34429 C1N5AS 10236295 EC50 = 81 nM T34429 C7L5PB 10246574 Ki = 500 nM T34429 CJ1E4U 10263398 EC50 > 100000 nM T34429 CX8B5S 10267729 Ki = 6.9 nM T34429 CMNH04 10286136 Ki = 1 nM T34429 CKOE15 10291446 Ki = 1.8 nM T34429 CLC49H 10421899 Ki = 8000 nM T34429 CHR72Q 10443815 Ki = 7900 nM T34429 CLDM93 10445840 Ki = 12.5 nM T34429 C92GSC 10471289 IC50 = 209000 nM T34429 CO6C5U 10472207 Ki >= 31622.78 nM T34429 CAKM87 10476928 Ki = 25.7 nM T34429 CPQ7O4 10560219 Ki > 10000 nM T34429 C61LSF 10560220 Ki > 10000 nM T34429 C1SFD2 10702168 Ki = 1275 nM T34429 CM0YS3 10799899 EC50 > 10000 nM T34429 CN0JI4 10911949 IC50 > 100000 nM T34429 CJM0E5 10924232 EC50 = 10964.78 nM T34429 CZR3T6 10932563 IC50 = 1600 nM T34429 CLD5Z0 11098414 IC50 = 27000 nM T34429 CD2H5V 11106445 EC50 > 100000 nM T34429 C0X9JF 11162968 Ki = 0.24 nM T34429 CO83JA 11183894 IC50 = 7400 nM T34429 CA0F6Z 11311114 Ki = 30.3 nM T34429 CC9Q3V 11332920 Ki = 100000 nM T34429 C08TAW 11458897 Ki = 3162.28 nM T34429 CP1WH5 11461365 EC50 = 2200 nM T34429 CYG3H9 11543786 Ki = 2.1 nM T34429 C72MKH 11581017 IC50 = 55000 nM T34429 C9GV3E 11673094 EC50 > 100000 nM T34429 CN4Z5C 11679149 EC50 = 100 nM T34429 CIQ12L 11701287 Ki = 399 nM T34429 C3M8DW 11709098 Ki = 3.2 nM T34429 CQ2Z8J 11738788 Ki = 8.3 nM T34429 CU08KY 11838799 EC50 = 10000 nM T34429 CB34AR 11957729 EC50 = 280 nM T34429 CDPE69 11983345 Ki = 1.3 nM T34429 C4MGN0 12272373 IC50 = 100000 nM T34429 CF96QD 12303261 IC50 = 4640 nM T34429 CLJ14R 12358972 IC50 = 1200 nM T34429 C4W6QV 12621483 EC50 = 7500 nM T34429 CE5X1A 12625600 Ki = 430 nM T34429 C5T1AQ 12752005 Ki >= 31622.78 nM T34429 CV1P7Z 13076422 Ki >= 31622.78 nM T34429 C5UK2P 13996231 Ki > 100000 nM T34429 C17ZBV 14262870 Ki = 10000 nM T34429 C6EO2H 14262872 Ki = 18000 nM T34429 C7HLF0 14539367 Ki = 398.11 nM T34429 CFCR71 15462089 EC50 = 9500 nM T34429 CW09EN 15557180 EC50 = 9000 nM T34429 C2EY3S 16210745 Ki = 3981.07 nM T34429 CGZN70 16637618 Ki = 2000 nM T34429 CJ7MZ2 16725873 EC50 = 1300 nM T34429 C9O4RE 16727410 Ki = 818 nM T34429 C3W8ZK 17758335 Ki = 1995.26 nM T34429 COF61U 17982621 Ki = 14.6 nM T34429 C1OTB6 18177037 Ki = 34000 nM T34429 C0KHB3 18180543 Ki = 524.5 nM T34429 C1WG4X 18180586 Ki = 268.4 nM T34429 C6K8VH 20754424 EC50 = 182 nM T34429 CCO62K 21124461 Ki = 1000 nM T34429 CQ03LX 21290600 IC50 = 1000 nM T34429 C0EO2W 22215312 Ki = 10000 nM T34429 C90DNQ 23599502 Ki = 26.9 nM T34429 CW2R4M 23624283 EC50 = 50.12 nM T34429 CYQ04C 23652627 Ki = 11.6 nM T34429 C8NKG4 23729371 IC50 = 6010 nM T34429 CHNO56 23729420 IC50 = 170 nM T34429 CU72MV 23729443 IC50 = 8.8 nM T34429 CCK0E4 23729447 IC50 = 91 nM T34429 CZ3Y2I 24743361 IC50 = 1510 nM T34429 C8ELU9 24782303 EC50 = 199.53 nM T34429 CJ6SF5 24782306 EC50 = 316.23 nM T34429 C01UNQ 24782307 EC50 = 199.53 nM T34429 C7KB8R 24782550 EC50 = 100 nM T34429 C3VF5D 24782552 EC50 = 158.49 nM T34429 C1BQK0 24782553 EC50 = 398.11 nM T34429 CSPX91 24782554 EC50 = 1995.26 nM T34429 C7A8DI 24782800 EC50 = 3162.28 nM T34429 C5TOI2 24782801 EC50 = 1258.93 nM T34429 C7FZ2J 24782802 EC50 = 125.89 nM T34429 C8S4LC 24782803 EC50 = 125.89 nM T34429 C4KT6W 24782804 EC50 = 199.53 nM T34429 C2IXL5 24782805 EC50 = 31.62 nM T34429 CDEB17 24783056 EC50 = 15.85 nM T34429 C3J4RX 24785333 EC50 = 501.19 nM T34429 CMPH82 24785597 EC50 = 63.1 nM T34429 C7HI4R 24785600 EC50 = 251.19 nM T34429 CV7WH3 24785604 EC50 = 398.11 nM T34429 CTF93A 24785864 EC50 = 251.19 nM T34429 C1JX7P 24785870 EC50 = 1000 nM T34429 CRD90F 24786134 EC50 = 158.49 nM T34429 C8E6VG 24786136 EC50 = 3981.07 nM T34429 C7K1EU 24786138 EC50 = 199.53 nM T34429 C69MBX 24786140 EC50 = 5011.87 nM T34429 CE2XP4 24795080 Ki = 6700 nM T34429 CD8JL5 24823533 EC50 > 100000 nM T34429 CO17TC 24833897 Ki = 198 nM T34429 CIR64L 24860582 EC50 = 3000 nM T34429 C38HOI 24876960 IC50 > 5000 nM T34429 C2YF8C 24877085 IC50 = 19 nM T34429 CH3OR9 24878344 IC50 = 11 nM T34429 CZD45C 24894145 EC50 > 100000 nM T34429 CIT85P 24894220 EC50 > 30000 nM T34429 C1QMI7 24894221 EC50 = 2600 nM T34429 CP91CV 24894236 EC50 > 30000 nM T34429 C9MSJ5 24894238 EC50 > 30000 nM T34429 C16LBC 24894240 EC50 > 30000 nM T34429 C4J3PZ 24894343 EC50 > 30000 nM T34429 CH1RI8 24894344 EC50 = 9400 nM T34429 CE6GL2 24894345 EC50 > 30000 nM T34429 C1HNK3 24894347 EC50 = 3600 nM T34429 CZ36RF 24895703 EC50 = 2600 nM T34429 CIDL67 24895833 EC50 > 30000 nM T34429 C3IL2C 24895834 EC50 = 4880 nM T34429 C85YMZ 24895835 EC50 = 4900 nM T34429 C7HJV0 24895836 EC50 > 30000 nM T34429 C84AQE 24945028 Ki = 5900 nM T34429 CHY7C1 24945029 Ki = 3700 nM T34429 CV07CE 24945030 Ki = 8200 nM T34429 C30XMU 24945031 Ki = 2600 nM T34429 CGI46H 24945032 Ki = 6300 nM T34429 C50QZG 24945033 Ki > 10000 nM T34429 CT13LF 24945123 Ki = 100000 nM T34429 CI0YH2 24945124 Ki = 14000 nM T34429 C3WIQ9 24945126 Ki = 7600 nM T34429 C93SUY 24945129 Ki = 19000 nM T34429 C5MNT9 24945296 Ki = 15000 nM T34429 C78HXO 24945297 Ki = 8200 nM T34429 CY5D6P 24945298 Ki > 10000 nM T34429 C1T0FO 24945299 Ki > 10000 nM T34429 C3UP8T 24945300 Ki > 10000 nM T34429 CKJG57 24945301 Ki > 10000 nM T34429 CW9F1R 24945302 Ki > 10000 nM T34429 C0N7YV 24945376 Ki > 10000 nM T34429 C3LBH5 24945542 Ki > 10000 nM T34429 CRYT93 24970319 Ki = 13000 nM T34429 C1XDF6 25009381 Ki = 28.84 nM T34429 CQR84M 25147644 Ki = 1 nM T34429 CI1V6B 25155668 Ki = 8.4 nM T34429 C9U2QX 25156769 Ki = 9.6 nM T34429 C6XVY0 25177374 Ki = 2290.87 nM T34429 CCB91S 25182691 Ki = 0.9 nM T34429 CF4OQ9 25182692 Ki = 3 nM T34429 C1CWU0 42631007 EC50 = 10 nM T34429 CFU84B 42636894 IC50 = 1730 nM T34429 CJO2D8 44138574 EC50 = 1200 nM T34429 CSEK38 44140519 EC50 = 10500 nM T34429 CJMB16 44140520 EC50 = 3900 nM T34429 CJV6A7 44158944 IC50 = 185 nM T34429 CXE4A6 44159538 IC50 = 99 nM T34429 C7BU8N 44190125 EC50 = 4470 nM T34429 CR80FS 44190223 EC50 > 100000 nM T34429 CB4K5O 44190326 EC50 > 100000 nM T34429 C83NGA 44190552 EC50 = 1150 nM T34429 C6NT5U 44190553 EC50 = 4260 nM T34429 C6TOC5 44199430 Ki = 4000 nM T34429 C43GIX 44222896 Ki = 1600 nM T34429 CBP9G1 44222951 Ki = 20 nM T34429 C6MCF2 44223074 Ki = 840 nM T34429 CG5Q6P 44223132 Ki = 3300 nM T34429 CCW0G6 44225415 Ki = 4.98 nM T34429 C4W0SH 44247585 Ki = 1.3 nM T34429 CJ2M9Q 44299190 Ki = 9.7 nM T34429 CY59RW 44348968 Ki = 13 nM T34429 CRC25U 44354684 EC50 = 19600 nM T34429 C1BC3P 44389116 Ki ~ 1000000 nM T34429 C1H7FD 44398087 IC50 = 9.6 nM T34429 C4E6XJ 44398088 IC50 = 61 nM T34429 C5L7UK 44398089 IC50 = 200 nM T34429 CH01FP 44398090 IC50 = 441 nM T34429 CNL4B1 44398091 IC50 = 0.75 nM T34429 C1C3EN 44398092 IC50 = 1.5 nM T34429 CF7HA2 44398095 EC50 = 44000 nM T34429 C2K1WB 44398115 IC50 = 14700 nM T34429 CYOE97 44399319 Ki = 5100 nM T34429 C3C2TD 44402933 Ki = 121.2 nM T34429 C20ZGN 44402935 Ki = 4.1 nM T34429 C1APT8 44402939 Ki = 1.1 nM T34429 CG9Y5H 44408892 Ki = 5011.87 nM T34429 COX8D7 44408895 Ki = 1258.93 nM T34429 CR6CE1 44408940 Ki = 2900 nM T34429 C9NW0H 44421540 Ki > 700 nM T34429 CPVN46 44421543 Ki > 700 nM T34429 CF73HK 44421545 Ki > 200 nM T34429 C20KPD 44423688 Ki = 15000 nM T34429 CYG93V 44427853 Ki = 1000 nM T34429 C3C2OK 44427854 Ki = 199.53 nM T34429 C8Y9FW 44427856 Ki = 50.12 nM T34429 C19LSU 44427858 Ki = 30 nM T34429 C1FY4M 44427860 Ki = 100 nM T34429 CC2BE1 44427862 Ki = 251.19 nM T34429 CW95BM 44427864 Ki = 590 nM T34429 C3XJ4Z 44427866 Ki = 199.53 nM T34429 C84GXL 44427868 Ki = 59 nM T34429 C8CPX2 44427870 Ki = 251.19 nM T34429 CS17TJ 44427872 Ki = 18 nM T34429 C5JU1B 44427874 Ki = 316.23 nM T34429 CDL67C 44427876 Ki = 1200 nM T34429 C9B6ER 44427877 Ki = 620 nM T34429 C15UHM 44427879 Ki = 230 nM T34429 CCAV10 44427881 Ki = 199.53 nM T34429 CXRV71 44427883 Ki = 98 nM T34429 CKX81C 44427885 Ki = 1584.89 nM T34429 CUR6V1 44430798 EC50 = 1500 nM T34429 C1JNK4 44442621 IC50 = 5200 nM T34429 C7WOJ8 44442623 IC50 = 4100 nM T34429 C1UES6 44448520 EC50 = 430 nM T34429 CJH2Y5 44448558 EC50 = 70 nM T34429 CM8U6J 44570006 Ki = 1000000 nM T34429 CH84MQ 44570007 Ki = 1000000 nM T34429 C2E3LJ 44570008 Ki = 1000000 nM T34429 CWPR65 44570009 Ki < 1000000 nM T34429 C13RLY 44570010 Ki < 1000000 nM T34429 CIV69B 44570011 Ki > 1000000 nM T34429 CG4YE9 44570012 Ki < 1000000 nM T34429 C0ZL8N 44570053 Ki > 1000000 nM T34429 CQ4K3T 44570054 Ki < 1000000 nM T34429 CVGP31 44570055 Ki < 1000000 nM T34429 CPST94 44570056 Ki > 1000000 nM T34429 C0VZ9I 44570057 Ki > 1000000 nM T34429 CQ8L9B 44570097 Ki > 1000000 nM T34429 CU7S2P 44570098 Ki > 1000000 nM T34429 CFUE82 44570099 Ki > 1000000 nM T34429 C31CSH 44570100 Ki > 1000000 nM T34429 CQS02B 44570101 Ki > 1000000 nM T34429 CMP1K2 44570102 Ki = 1000000 nM T34429 C2X4GC 44570103 Ki = 1000000 nM T34429 C18JSV 44570104 Ki < 1000000 nM T34429 C7I6OB 44570105 Ki = 1000000 nM T34429 C1A2TU 44575473 Ki = 1 nM T34429 CDX2H1 44621189 EC50 = 10000 nM T34429 C5N9PS 44719858 Ki >= 31622.78 nM T34429 CXYK56 45268365 Ki = 739 nM T34429 CQK28Z 45379093 Ki = 130 nM T34429 CS9A3Z 45484395 EC50 = 350 nM T34429 CO9R7V 46225140 EC50 = 9360 nM T34429 C50QER 46225183 EC50 = 11770 nM T34429 C3Y0MF 46225231 EC50 > 100000 nM T34429 C91OTQ 46225232 EC50 = 12900 nM T34429 C6XSL7 46830771 EC50 = 120 nM T34429 CL98UY 46831060 EC50 = 130 nM T34429 CE71GL 46846404 Ki = 2.5 nM T34429 CQ8KI6 46878168 EC50 = 25000 nM T34429 CZ0A7U 46890769 EC50 = 11000 nM T34429 C1AK8C 46890770 EC50 = 12000 nM T34429 CB6T3M 46890771 EC50 = 1500 nM T34429 CP8FW2 46890772 EC50 = 540 nM T34429 CX7I3Y 46890773 EC50 = 12000 nM T34429 C2I9CM 46890824 EC50 = 2100 nM T34429 C6RB1V 46890825 EC50 = 3200 nM T34429 C5JT1D 46890826 EC50 = 7400 nM T34429 CC0E7P 46890827 EC50 = 27000 nM T34429 CT6UY7 46890828 EC50 = 33000 nM T34429 C9QFU5 46890891 EC50 = 800 nM T34429 CS74RA 46890892 EC50 = 700 nM T34429 CNQ26O 46890893 EC50 = 18000 nM T34429 CZQ25U 46890894 EC50 = 4600 nM T34429 CJ8YV7 46890895 EC50 = 1800 nM T34429 CWDG43 46890952 EC50 = 4700 nM T34429 CIC32L 46890953 EC50 = 5300 nM T34429 C4ZYM8 46890954 EC50 = 300 nM T34429 C0P4GM 46890955 EC50 = 1000 nM T34429 CK94BQ 46890956 EC50 = 2800 nM T34429 CEW98A 46891012 EC50 = 3900 nM T34429 C3CPE9 46891013 EC50 = 1600 nM T34429 C51IBN 46891527 EC50 = 2700 nM T34429 CQ34CV 46891528 EC50 = 1500 nM T34429 CH91DV 46891529 EC50 = 1100 nM T34429 C7LS0J 46891530 EC50 = 900 nM T34429 CCE34G 46891585 EC50 = 1200 nM T34429 CMJ93X 46891586 EC50 = 2700 nM T34429 CHGA57 46891587 EC50 = 1700 nM T34429 C2FOK8 46891588 EC50 = 400 nM T34429 C4ZXM7 46891589 EC50 = 5600 nM T34429 CK9NM5 46935872 Ki = 413 nM T34429 CGS59I 49780184 Ki = 38.9 nM T34429 C8BL3Y 49780185 Ki = 109.65 nM T34429 CXC71P 49780186 Ki = 43.65 nM T34429 C2UE4C 49780187 Ki = 6918.31 nM T34429 C0AZL7 49780189 Ki = 3311.31 nM T34429 CRQ28M 49783248 Ki = 18.62 nM T34429 C8QR3T 49783249 Ki = 2.692 nM T34429 CQF5Z0 49783448 Ki = 61.66 nM T34429 C2AWC6 49783449 Ki = 6 nM T34429 C1HN5U 49783450 Ki = 43.65 nM T34429 C2X5HQ 49783451 Ki = 37.15 nM T34429 CMJ1K8 49837893 Ki = 11.6 nM T34429 C5TH3U 49859909 EC50 > 316227.77 nM T34429 CR53VH 49862169 Ki = 3300 nM T34429 C15OJH 49862213 Ki > 15000 nM T34429 CT3WH4 49862215 Ki = 1580 nM T34429 C15JDC 49862217 Ki > 15000 nM T34429 CT39UZ 49862259 Ki > 13500 nM T34429 CHBT02 49862263 Ki > 15000 nM T34429 C47WAJ 49862265 Ki = 7590 nM T34429 CV96ZG 49862267 Ki = 4750 nM T34429 CQ38SD 49862303 Ki > 15000 nM T34429 CL7KG5 49862305 Ki = 9870 nM T34429 C9G7LW 49862307 Ki = 14600 nM T34429 CGI23Z 49862361 Ki > 15000 nM T34429 CAI26L 49862363 Ki > 15000 nM T34429 CC1SF7 49863118 EC50 = 1.995 nM T34429 CN93ZT 49863119 EC50 = 1.995 nM T34429 C05BDV 49863120 EC50 = 3.162 nM T34429 C2R3SE 49863121 EC50 = 10 nM T34429 CU5A7B 49863149 EC50 = 6.31 nM T34429 C7FET8 49863150 EC50 = 7.943 nM T34429 CW96TD 49863151 EC50 = 10 nM T34429 CTP40J 49863152 EC50 = 10 nM T34429 CHSG10 49863184 EC50 = 31.62 nM T34429 CL8SE4 49863185 EC50 = 25.12 nM T34429 CVJ27M 49863186 EC50 = 25.12 nM T34429 CSKG13 49863187 EC50 = 25.12 nM T34429 C5R4PV 53245679 Ki = 5011.87 nM T34429 C3AKS2 53302872 Ki = 221 nM T34429 CFK71X 53319046 IC50 = 7000 nM T34429 C8PN4O 53321089 IC50 = 7200 nM T34429 C0YJH8 53321777 Ki = 57 nM T34429 CQ2BW7 53322415 IC50 = 6100 nM T34429 C8L2WR 53322955 IC50 = 5600 nM T34429 CJ3D7I 53483934 IC50 > 10000 nM T34429 CJ34EQ 53483935 IC50 = 4600 nM T34429 CA6B7M 54580336 IC50 = 1190 nM T34429 CK32EN 54601756 EC50 = 5400 nM T34429 CE7WZ8 54754345 Ki >= 31622.78 nM T34429 C7E9TR 56589586 EC50 = 25703.96 nM T34429 C8DO6C 56594103 EC50 = 5754.4 nM T34429 C6QHA3 56594105 EC50 = 20892.96 nM T34429 CVHC26 56594107 EC50 = 29512.09 nM T34429 CID40G 56594247 EC50 = 7762.47 nM T34429 C7AM2S 56594249 EC50 = 20417.38 nM T34429 CQO86Z 56594251 EC50 = 9772.37 nM T34429 CGP37R 56594253 EC50 = 44668.36 nM T34429 CNP6K0 56594255 EC50 = 4786.3 nM T34429 CLH24J 56663402 IC50 > 10000 nM T34429 CS10RB 56663482 EC50 = 10000 nM T34429 C3ZOB8 56663483 Ki >= 31622.78 nM T34429 CU7OP3 56666825 IC50 > 10000 nM T34429 CY01LS 56666826 IC50 > 10000 nM T34429 CCP40B 56666827 IC50 > 10000 nM T34429 C4XE6O 56666905 Ki = 10000 nM T34429 C4O6ID 56666906 Ki >= 31622.78 nM T34429 CZF26A 56666907 EC50 = 10000 nM T34429 CVT85Q 56670262 IC50 > 10000 nM T34429 CBJS01 56670295 Ki >= 31622.78 nM T34429 CP9WN5 56673804 EC50 = 10000 nM T34429 CPO8M4 56675778 EC50 = 1862.09 nM T34429 CN0AZ3 56677030 Ki >= 31622.78 nM T34429 C7XK8I 56677105 IC50 = 15100 nM T34429 C02AZR 56677106 IC50 > 10000 nM T34429 CUIY40 56679246 IC50 = 3300 nM T34429 CF76SY 56680450 Ki = 19952.62 nM T34429 C7L2JC 56680506 Ki >= 31622.78 nM T34429 C0Z8XY 56680507 Ki >= 31622.78 nM T34429 CY70FV 56941220 EC50 = 1200 nM T34429 C4GSE6 57329546 EC50 = 180 nM T34429 CEG4N8 57334716 EC50 > 100000 nM T34429 CNB85W 57391663 Ki = 6309.57 nM T34429 CCVI85 57391664 Ki = 12589.25 nM T34429 CX48RS 57391706 Ki = 12589.25 nM T34429 C63HMW 57393442 Ki = 25118.86 nM T34429 C4WDS2 57396902 Ki = 19952.62 nM T34429 CPO50Z 57397665 Ki = 1584.89 nM T34429 C0PCS9 57398597 Ki = 12589.25 nM T34429 C3YVT8 57398685 Ki = 10000 nM T34429 CA1LW2 57400332 Ki = 39810.72 nM T34429 CV31DZ 57485530 Ki = 4 nM T34429 CZ4G2Y 57485620 Ki = 19 nM T34429 C9G5JE 57485797 Ki = 105 nM T34429 CR2V6D 57485798 Ki = 3220 nM T34429 CG1TP6 57485799 Ki = 22 nM T34429 CON1Z4 57485800 Ki = 4.6 nM T34429 CDW7N1 57486266 Ki = 1849 nM T34429 CCM98N 57486336 Ki = 39 nM T34429 CVL35M 57521318 IC50 = 40000 nM T34429 C6M5EA 57521710 IC50 = 6900 nM T34429 C5PG6A 57523184 IC50 = 5000 nM T34429 CB71LF 57523367 IC50 = 45000 nM T34429 CJYS25 57663369 EC50 = 316.23 nM T34429 C4QG8R 57663382 EC50 = 63.1 nM T34429 CHQI67 57663405 EC50 = 63.1 nM T34429 CA9RK8 57663418 EC50 = 630.96 nM T34429 CM7H9G 57663419 EC50 = 501.19 nM T34429 C58ERT 57663421 EC50 = 100 nM T34429 CY2S7K 57663434 EC50 = 39.81 nM T34429 C9A0XM 57663447 EC50 = 100 nM T34429 C18FHN 57663450 EC50 = 15.85 nM T34429 CPSX03 57663451 EC50 = 251.19 nM T34429 CMUD63 57663495 EC50 = 199.53 nM T34429 CVL35Z 57663496 EC50 = 31.62 nM T34429 CBK0Y1 57663581 EC50 = 794.33 nM T34429 CSK82C 57663586 EC50 = 19.95 nM T34429 C5J1QT 57663596 EC50 = 100 nM T34429 CTV29J 57663598 EC50 = 63.1 nM T34429 C2X7OT 57663610 EC50 = 100 nM T34429 C98CVM 57663630 EC50 = 79.43 nM T34429 CGA1V2 57663637 EC50 = 3162.28 nM T34429 CV2J9A 57663655 EC50 = 125.89 nM T34429 CR7S5U 57663666 EC50 = 251.19 nM T34429 C4GXF1 57663688 EC50 = 50.12 nM T34429 C9IU7S 58081849 EC50 = 41 nM T34429 C7O3GZ 58088026 EC50 = 63 nM T34429 CND4G1 58088117 EC50 = 45 nM T34429 CP15TC 58201402 Ki = 300 nM T34429 CW03VZ 58201405 Ki = 1400 nM T34429 CP47JL 58201407 Ki = 6900 nM T34429 CMKN28 58201409 Ki = 10 nM T34429 CP8G5N 58201418 Ki = 2700 nM T34429 C0TML6 58201419 Ki = 100 nM T34429 CB32IW 58201420 Ki = 990 nM T34429 CRC51J 58201424 Ki = 400 nM T34429 C2XCI7 58312740 Ki = 20000 nM T34429 C3KJ7N 58488107 Ki = 350 nM T34429 COQ52A 59268918 Ki > 10000 nM T34429 C4S7VM 59268924 Ki > 10000 nM T34429 CYV48O 59268925 Ki = 1200 nM T34429 C4N2FX 59268932 Ki = 4700 nM T34429 CSW42A 59268935 Ki > 10000 nM T34429 CVN48B 59268936 Ki > 10000 nM T34429 CYSC50 59268939 Ki > 10000 nM T34429 CTR7E8 59268940 Ki > 10000 nM T34429 CHR48L 59268945 Ki = 5900 nM T34429 C1TJ6W 59268948 Ki > 10000 nM T34429 C3EJ6I 59268964 Ki = 4600 nM T34429 CT61RD 59268965 Ki > 10000 nM T34429 C9OS6X 59361675 Ki = 1300 nM T34429 C1J5PV 59361705 Ki = 7800 nM T34429 C68WRJ 59403312 Ki = 27000 nM T34429 C6OJH7 59403341 Ki = 3400 nM T34429 CHFI16 60167958 EC50 = 324 nM T34429 CX90RF 66211794 Ki = 100000 nM T34429 CXN68J 66212381 Ki = 20000 nM T34429 C65UFK 66213161 Ki = 100000 nM T34429 C79SIL 66796791 IC50 = 6 nM T34429 C9BF6L 66797369 EC50 = 200 nM T34429 C4S0IK 67144490 Ki = 31 nM T34429 CRSX31 68024489 Ki > 10000 nM T34429 CPA38K 68024616 Ki = 8800 nM T34429 CGU14E 68024620 Ki > 10000 nM T34429 C38FDK 68024820 Ki > 10000 nM T34429 CR0Q4N 68465506 Ki = 140 nM T34429 CSR1I4 69249623 EC50 = 1570 nM T34429 CF9TX0 69604735 Ki > 300 nM T34429 CN1T4U 69925573 EC50 = 180 nM T34429 CE0N4K 70675110 Ki = 174.5 nM T34429 CO5RQ6 70692779 IC50 = 10000 nM T34429 CJX80U 71201914 EC50 = 670 nM T34429 C4SQ8J 71201919 EC50 = 5800 nM T34429 C2TLN3 71201939 EC50 = 390 nM T34429 CU0I5B 71201952 EC50 = 2000 nM T34429 CV42PL 71201953 EC50 = 790 nM T34429 CB4Q0O 71299322 Ki = 0.24 nM T34429 C6LM4P 71449313 Ki = 2511.89 nM T34429 C0DX3I 71449982 Ki = 1421 nM T34429 C5BH6L 71450029 Ki = 8006 nM T34429 CQE53F 71450030 Ki = 39 nM T34429 C96JMX 71450130 Ki = 8200 nM T34429 CZCT16 71450152 Ki = 2156 nM T34429 C4W9AV 71450153 Ki = 24.1 nM T34429 C60AXY 71450154 Ki = 60 nM T34429 C1HN0O 71450156 Ki = 2027 nM T34429 CS3N9F 71450157 Ki = 705 nM T34429 CV9CO0 71450158 Ki = 4.5 nM T34429 C2I4CF 71450171 Ki = 210 nM T34429 CZJ5S3 71451115 Ki = 1584.89 nM T34429 CRX2E6 71451808 Ki = 6530 nM T34429 CQ5XI6 71451809 Ki = 590 nM T34429 C9J0NM 71451810 Ki = 1.2 nM T34429 C5SX4G 71451811 Ki > 10000 nM T34429 CZ42AI 71451812 Ki = 3.3 nM T34429 CB6V1U 71451813 Ki = 15 nM T34429 C9DH7V 71451944 Ki = 13000 nM T34429 CL2A9E 71451983 Ki = 240 nM T34429 C2BGU6 71451984 Ki = 6.2 nM T34429 CA69ND 71451985 Ki = 1097 nM T34429 CADC24 71451986 Ki = 2.1 nM T34429 CJ01HW 71451994 Ki = 40 nM T34429 C7AFY5 71452017 Ki = 352 nM T34429 C70RFX 71452018 Ki = 36.1 nM T34429 C3EZ1O 71453019 IC50 = 1.09 nM T34429 CI8YM0 71453627 Ki = 7.2 nM T34429 C1OS8W 71453628 Ki = 330 nM T34429 C89KME 71453629 Ki = 641 nM T34429 CDGO46 71453630 Ki = 79 nM T34429 C3UW8E 71453631 Ki = 70 nM T34429 C91CNU 71453666 Ki = 13 nM T34429 CV0Q4C 71453769 Ki = 8600 nM T34429 CJL26M 71453770 Ki = 14000 nM T34429 CJ1RO8 71453794 Ki = 15 nM T34429 C7JGE0 71453795 Ki = 6.4 nM T34429 CQ0W3F 71453796 Ki = 52.5 nM T34429 CE7U4Q 71453797 Ki = 2.8 nM T34429 C2HS8T 71453798 Ki = 5.9 nM T34429 CKHF18 71453822 Ki = 5.5 nM T34429 CI8RM2 71453823 Ki = 29 nM T34429 CE96BS 71455355 Ki = 30 nM T34429 CLX57K 71455356 Ki = 74 nM T34429 CNGK53 71455357 Ki = 605 nM T34429 C8N4IJ 71455358 Ki = 4545 nM T34429 CDC54A 71455359 Ki = 1007 nM T34429 C8Z4ES 71455499 Ki = 100000 nM T34429 CFOH06 71455500 Ki = 14000 nM T34429 CT79WZ 71455501 Ki = 14000 nM T34429 CSK73V 71455528 Ki = 20 nM T34429 C71PCM 71455535 Ki = 5500 nM T34429 CSR6I8 71455553 Ki = 2.2 nM T34429 CN31FI 71455554 Ki = 259 nM T34429 CFMS41 71457131 Ki > 10000 nM T34429 C18UJA 71457132 Ki = 4847 nM T34429 CO5B7Z 71457133 Ki = 20 nM T34429 CK10DR 71457134 Ki = 1.3 nM T34429 CCFH76 71457135 Ki = 17 nM T34429 CY4U7W 71457136 Ki = 3.6 nM T34429 CDQ91P 71457319 Ki = 46 nM T34429 CS8ZC6 71457320 Ki = 1803 nM T34429 CY54OR 71457321 Ki = 961 nM T34429 CO5Z7A 71457322 Ki = 30 nM T34429 CZDF62 71457323 Ki = 22.1 nM T34429 CFW9G2 71457348 Ki = 1.8 nM T34429 CGYS73 71457349 Ki = 11.5 nM T34429 CN0AH1 71458995 Ki = 77 nM T34429 C7V0CY 71458996 Ki > 10000 nM T34429 CH7U6N 71458997 Ki = 43.9 nM T34429 CUC0T8 71458998 Ki = 1.6 nM T34429 C96NIY 71459035 Ki = 73 nM T34429 C1WME8 71459126 Ki = 1600 nM T34429 C3IJ1A 71459152 Ki = 150 nM T34429 C5IAT7 71459153 Ki = 94 nM T34429 C4S9BP 71459154 Ki = 4.3 nM T34429 CP1M7A 71459155 Ki = 1.1 nM T34429 CB4M3E 71459156 Ki = 0.51 nM T34429 C3B7PW 71459157 Ki = 0.8 nM T34429 C8IVG6 71459158 Ki = 11.2 nM T34429 CH9QF6 71459203 Ki = 4.7 nM T34429 CW2YF0 71459204 Ki = 15.7 nM T34429 CU5D0T 71460792 Ki = 1305 nM T34429 CW58SI 71460793 Ki = 80 nM T34429 CU7CZ6 71460794 Ki > 10000 nM T34429 CZKD91 71460795 Ki = 7565 nM T34429 CWJ1I2 71460832 Ki = 160 nM T34429 C0G4SZ 71460833 Ki = 13 nM T34429 C5TSZ4 71460834 Ki = 23 nM T34429 C69UGX 71460958 Ki = 76 nM T34429 CH57RZ 71460959 Ki = 5.9 nM T34429 C1UP7D 71460960 Ki = 3.8 nM T34429 COH7P4 71460982 Ki = 5 nM T34429 CZO67H 71460983 Ki = 12.3 nM T34429 C7AQS1 71460984 Ki = 33.8 nM T34429 CV37ZJ 71462520 Ki = 23 nM T34429 C86IYC 71462521 Ki > 10000 nM T34429 CFD1B9 71462522 Ki = 281 nM T34429 C3YZ6W 71462523 Ki = 33 nM T34429 CK3N6Z 71462524 Ki = 111.4 nM T34429 C1MKL2 71462677 Ki = 851 nM T34429 C2EU1R 71462678 Ki = 219 nM T34429 CU93PT 71462679 Ki = 168 nM T34429 CLS59K 71462680 Ki = 66.2 nM T34429 C1V0ZI 71462681 Ki = 56.3 nM T34429 C6D0TN 71462682 Ki = 87.7 nM T34429 CZW76V 71462683 Ki = 1.2 nM T34429 CM0HG2 71462689 Ki = 560 nM T34429 CG7ZE8 71462717 Ki = 59 nM T34429 CJ7ER8 71682669 Ki = 4500 nM T34429 C05CTI 71682670 Ki = 350 nM T34429 CMKP08 71682671 Ki = 1900 nM T34429 CT34ZA 71682672 Ki = 100000 nM T34429 CE50MN 71682827 Ki = 15000 nM T34429 C9C3EG 71682975 Ki = 10000 nM T34429 C20NXV 71682976 Ki = 11000 nM T34429 CTN89W 71713941 IC50 = 41000 nM T34429 CINY69 72192461 EC50 = 35 nM T34429 CSW89Y 72709023 EC50 = 880 nM T34429 CQ30RG 72709025 EC50 > 10000 nM T34429 C9AD0M 72709102 EC50 = 990 nM T34429 C0JXT9 72709105 EC50 = 26 nM T34429 C6QOL9 72709106 EC50 = 170 nM T34429 C12AOM 72709107 EC50 = 1200 nM T34429 C48SNQ 72709187 EC50 = 290 nM T34429 CA2BX4 72709190 EC50 = 1300 nM T34429 CA94ZJ 72709267 EC50 = 530 nM T34429 CXA2P7 72709272 EC50 = 56 nM T34429 CNGR78 72709273 EC50 = 550 nM T34429 CH2RT8 72709349 EC50 = 490 nM T34429 C1K9OD 72709587 EC50 = 150 nM T34429 COH37Y 72709588 EC50 = 120 nM T34429 CZB6J7 72709589 EC50 = 750 nM T34429 CLM6P9 72709673 EC50 = 53 nM T34429 CL01VG 72709675 EC50 = 140 nM T34429 CCM45B 72709679 EC50 = 62 nM T34429 CP52FZ 72709766 EC50 = 5600 nM T34429 C56HYB 72710014 EC50 = 1100 nM T34429 CBI45H 72711595 EC50 = 140 nM T34429 CNR89U 72711804 EC50 = 1900 nM T34429 CXN73A 72711809 EC50 = 130 nM T34429 CRK9B0 72712019 EC50 = 450 nM T34429 CX47HS 72712022 EC50 = 220 nM T34429 C3NZR4 72712025 EC50 = 560 nM T34429 CW4IE9 72712233 EC50 = 2500 nM T34429 CH8R3W 72712234 EC50 = 380 nM T34429 COGD09 72712235 EC50 = 160 nM T34429 CT50LG 72712451 EC50 = 3000 nM T34429 C2NTD8 72712453 EC50 = 210 nM T34429 C64JFG 72712456 EC50 = 4900 nM T34429 C1KT0W 73347339 Ki = 48700 nM T34429 C87TLQ 73347340 Ki = 10500 nM T34429 CY56RE 73347561 Ki = 100 nM T34429 CD8OT4 73348844 Ki = 4500 nM T34429 CL73CV 73350432 Ki = 1100 nM T34429 CEBL05 73350433 Ki = 29500 nM T34429 C71LER 73350667 Ki = 5 nM T34429 C5ILK3 73351944 Ki = 6700 nM T34429 CER79N 73352166 Ki = 300 nM T34429 CIX69R 73353186 IC50 = 5 nM T34429 CL6S2I 73353403 Ki = 29300 nM T34429 CYL5C0 73355120 Ki = 30 nM T34429 C5PJ4Z 73356479 Ki = 232000 nM T34429 C1LAP7 73759679 IC50 = 100000 nM T34429 CKD42Z 75113427 Ki = 5.4 nM T34429 C3CH5U 76310142 IC50 = 103 nM T34429 CF7TP2 76310143 IC50 = 4700 nM T34429 C1BA3C 76311214 IC50 = 2200 nM T34429 CT0N4Q 76311216 IC50 = 1300 nM T34429 CWG93E 76314835 IC50 = 2300 nM T34429 CFG3N4 76318436 IC50 = 2200 nM T34429 C0HEJ6 76321094 IC50 > 10000 nM T34429 C72USC 76322102 Ki = 600 nM T34429 CF5OB2 76324742 IC50 = 497 nM T34429 CQ4D8U 76325731 IC50 = 41300 nM T34429 C6S9CQ 76329290 IC50 = 3400 nM T34429 C5YE3Q 76332941 IC50 = 2200 nM T34429 CKZ19D 76336550 IC50 = 2000 nM T34429 CJ9N1O 76336552 IC50 = 2700 nM T34429 CPHO43 77907039 Ki = 72.8 nM T34429 CC4PX8 78210299 EC50 = 3300 nM T34429 C8PQY5 86272237 EC50 = 2140 nM T34429 C68SVO 86272238 EC50 = 9630 nM T34429 C1PU3W 86272239 EC50 = 4640 nM T34429 CMVG94 86272241 EC50 > 20000 nM T34429 CWY3H2 86272242 EC50 > 20000 nM T34429 C4X2HY 86272243 EC50 = 2490 nM T34429 CB40AF 86272489 EC50 = 3540 nM T34429 CX8EB0 86272490 EC50 = 3990 nM T34429 C28YBH 86272491 EC50 = 6920 nM T34429 CRN39M 86272492 EC50 > 20000 nM T34429 C8BKD7 86272493 EC50 = 10480 nM T34429 CP7N9X 86272494 EC50 = 4750 nM T34429 CSW3G7 86272495 EC50 > 20000 nM T34429 CY9D7R 86272718 EC50 > 20000 nM T34429 CTKH23 86272719 EC50 > 20000 nM T34429 CKUG03 86272720 EC50 > 20000 nM T34429 C1SP2V 86272721 EC50 > 20000 nM T34429 CCK2W0 86272722 EC50 > 20000 nM T34429 CLBP52 86272723 EC50 > 20000 nM T34429 C1X0MC 86275816 EC50 = 3980 nM T34429 C5V6AB 86275817 Ki = 14.9 nM T34429 CK3CP4 86275818 EC50 = 8380 nM T34429 CZCV56 89943572 Ki = 73 nM T34429 CUX53L 89943718 Ki = 117 nM T34429 CEI2S7 89943719 Ki = 133 nM T34429 C2HUL4 90659973 Ki = 1000 nM T34429 CEO8K1 90664654 Ki > 700 nM T34429 C6CK4V 90666446 Ki > 100000 nM T34429 CWO82R 90666447 Ki = 2187.76 nM T34429 C82BRL 90670746 Ki = 0.092 nM T34429 CDR3J6 118714573 EC50 = 8900 nM T34429 CMZY72 118714574 EC50 = 67000 nM T34429 CME75X 118714575 EC50 = 10700 nM T34429 C1LI5O 118714576 EC50 = 7300 nM T34429 CRN5W8 118714577 EC50 = 3900 nM T34429 COBN35 118714578 EC50 = 2600 nM T34429 C4Y2TK 118714579 EC50 = 1900 nM T34429 COU80J 118714972 IC50 = 2344.23 nM T34429 C8FL2V 118714973 IC50 = 590 nM T34429 CYJ4U2 118714975 IC50 = 3100 nM T34429 CA39EX 118714977 IC50 = 3300 nM T34429 C08XJQ 118714978 IC50 = 812.83 nM T34429 C1FM5W 118720625 IC50 = 4168.69 nM T34429 C2DCT5 118720627 IC50 = 21000 nM T34429 C3H4AX 118720665 IC50 = 3950 nM T34429 CR0P7N 122553341 Ki = 9.61 nM T34429 C2Q0DP 124121313 EC50 = 3200 nM T34429 CUPV95 124121322 EC50 = 2050 nM T34429 CI7F3J 124121346 EC50 = 2170 nM T34429 CW1H3O 124121348 EC50 = 5650 nM T34429 CZAG04 124121349 EC50 = 1260 nM T34429 CSH0L2 124121350 EC50 = 20430 nM T34429 C0UO2Q 124121352 EC50 = 6990 nM T34429 CH2Z0U 124121355 EC50 = 7650 nM T34429 CGKN64 124121356 EC50 = 3150 nM T34429 CZMO80 124121450 EC50 = 5020 nM T34429 C7BO3N 124121470 EC50 = 8450 nM T34429 CS6RL2 124121477 EC50 = 7650 nM T34429 CUCV59 124121482 EC50 = 8390 nM T34429 C3K0WD 124220259 EC50 = 500 nM T34429 CGE7M2 124220260 EC50 = 70 nM T34429 CVOQ45 127027055 EC50 = 60000 nM T34429 CHDL08 127030959 EC50 > 20000 nM T34429 C8NF2J 127031839 EC50 > 20000 nM T34429 CN7U5B 127032216 EC50 > 20000 nM T34429 C54QBL 127032221 EC50 > 20000 nM T34429 C35TXU 127032222 EC50 > 20000 nM T34429 CX0JE5 127032223 EC50 > 20000 nM T34429 CN3D9L 127032224 EC50 > 20000 nM T34429 C2JR0N 127032225 EC50 > 20000 nM T34429 CAMT80 127032420 EC50 = 8600 nM T34429 C3TQ0Z 127032514 EC50 > 20000 nM T34429 CSM4N5 127032515 EC50 > 20000 nM T34429 CCN6S3 127032516 EC50 > 20000 nM T34429 CMJ2L4 127032526 EC50 > 20000 nM T34429 CR45UW 127032527 EC50 > 20000 nM T34429 CV4Q1T 127032528 EC50 > 20000 nM T34429 C6FLK5 127032529 EC50 > 20000 nM T34429 CETJ16 127032702 EC50 > 20000 nM T34429 CYD92I 127032830 EC50 > 20000 nM T34429 COIT46 127032831 EC50 > 20000 nM T34429 CI6A3T 127032836 EC50 > 20000 nM T34429 C68WOD 127032837 EC50 > 20000 nM T34429 CB0DQ1 127033408 EC50 = 2830 nM T34429 CH0N1M 127033409 EC50 = 14130 nM T34429 CIO0D8 127034497 EC50 > 20000 nM T34429 CU6K4N 127034498 EC50 > 20000 nM T34429 CPCW81 127039568 EC50 = 1410 nM T34429 CK59DM 127039569 EC50 = 1090 nM T34429 C3NU4S 127043061 IC50 > 5000 nM T34429 CM8FN5 130448139 EC50 = 93 nM T34429 CG0CP8 130448165 EC50 = 110 nM T34429 CUIB45 130448288 EC50 = 69 nM T34429 C7U3RI 130448318 EC50 = 88 nM T34429 CUI37O 130448447 EC50 = 71 nM T34429 CA01US 130448674 EC50 = 98 nM T34429 CDW92O 130448691 EC50 = 83 nM T34429 CSV59E 134131673 EC50 = 4200 nM T34429 CL3IE5 134132150 EC50 = 320 nM T34429 CA4X5H 134133656 EC50 = 940 nM T34429 C6XCO7 134134094 EC50 = 410 nM T34429 CDSM51 134134865 EC50 = 260 nM T34429 CKB5T2 134136620 EC50 = 31 nM T34429 C3GH1V 134136714 EC50 = 120 nM T34429 C0JKY3 134138261 EC50 = 140 nM T34429 C03MJH 134139949 EC50 = 300 nM T34429 C1E2RC 134141899 EC50 = 40 nM T34429 CNK1L0 134142616 EC50 = 260 nM T34429 CXQ84A 134143789 EC50 = 91 nM T34429 C7AU1K 134146761 EC50 = 70 nM T34429 CD24RC 134150057 EC50 = 18 nM T34429 CH32TG 134153963 EC50 = 100 nM T34429 CA5O8R 134154723 EC50 = 41 nM T34429 CFY28D 134155678 EC50 = 95 nM T34429 CKB4X1 134157219 EC50 = 250 nM T34429 CLE38V 135508231 EC50 = 3000 nM T34429 CMC45A 137632866 EC50 = 5200 nM T34429 CFRE32 137633236 IC50 = 11000 nM T34429 CD0F1A 137636378 EC50 > 100000 nM T34429 CCL9R8 137637184 EC50 = 990 nM T34429 CN8Y4B 137637992 EC50 = 40000 nM T34429 CS2ID3 137638310 EC50 = 1600 nM T34429 C2PX0V 137639518 EC50 > 100000 nM T34429 CMHR69 137640337 EC50 = 2600 nM T34429 CMVI58 137642243 EC50 = 2200 nM T34429 C8BOJ1 137645300 EC50 = 5100 nM T34429 C1W5DC 137645588 Ki = 8000 nM T34429 CO6I0B 137645847 IC50 = 2000 nM T34429 C8XK9J 137647637 EC50 = 6500 nM T34429 C6MG4L 137647685 EC50 = 1200 nM T34429 CVU57Z 137650129 IC50 = 5700 nM T34429 C8W7ET 137650261 EC50 = 5400 nM T34429 CJS50P 137659552 Ki = 8000 nM T34429 CO1I0F 137660807 EC50 = 2600 nM T34429 CZE7W3 137661099 EC50 = 4400 nM T34429 C3FZL5 141725921 IC50 = 21.25 nM T34429 CIN05D 145968525 IC50 = 320 nM T34429 CTV32Z 145968583 IC50 > 1000 nM T34429 C24KCP 145979896 IC50 = 24.3 nM T34429 CG9QD6 145980121 Ki = 1930 nM T34429 C5UOR9 145980384 Ki = 909 nM T34429 C46QKG 145980538 EC50 = 93 nM T34429 CQX57J 145980876 EC50 = 98 nM T34429 CL5F4P 145981379 Ki = 559 nM T34429 C7AC3F 145984633 Ki = 1826 nM T34429 CDH85G 145986462 Ki = 617 nM T34429 C3U0HD 145986545 IC50 = 12.3 nM T34429 C0F1IT 145988882 Ki = 1288 nM T34429 C7XB0C 145989786 Ki = 4.4 nM T34429 C9U4IN 145989794 IC50 = 6.5 nM T34429 CYC3B7 145990104 Ki = 2800 nM T34429 C8V6DI 145990201 IC50 = 92 nM T34429 C0FL9I 145990275 IC50 = 47 nM T34429 CPI7X8 145990905 EC50 = 83 nM T34429 C74VEP 145991862 Ki = 984 nM T34429 CMY8S3 145991947 Ki = 1638 nM T34429 C6Q3XK 146680925 Ki = 33.2 nM T34429 C6DCN9 146680926 Ki = 660.5 nM T34429 CK5YB0 154734327 EC50 = 30 nM T34429 CC98US 155510766 IC50 = 196000 nM T34429 C9F6LV 155512339 Ki = 98.7 nM T34429 C97VTE 155512367 EC50 < 30000 nM T34429 CI7C6L 155513305 EC50 = 8270 nM T34429 CT64LK 155514460 Ki = 96.9 nM T34429 CF74UI 155514726 EC50 = 2500 nM T34429 CMV2G7 155515603 Ki = 149 nM T34429 C6F0WH 155515772 IC50 = 160000 nM T34429 C7DBH6 155516230 Ki = 74.9 nM T34429 CIN3J0 155517537 EC50 = 1350 nM T34429 CL8ED4 155517866 IC50 = 300000 nM T34429 C3TH5I 155517886 EC50 = 240 nM T34429 C86GDR 155518901 EC50 = 4960 nM T34429 CF31YA 155518951 IC50 = 12000 nM T34429 C15WRG 155519331 EC50 < 30000 nM T34429 CR6XT8 155519493 EC50 > 13300 nM T34429 C5GAS9 155521191 Ki = 279 nM T34429 CZO1K7 155521465 IC50 = 195000 nM T34429 CHC38D 155522533 Ki = 74.6 nM T34429 CK01QX 155522758 Ki = 29.3 nM T34429 CCD84W 155522888 EC50 = 110 nM T34429 CVI03B 155524051 EC50 = 2000 nM T34429 C4WLR1 155525465 EC50 = 140 nM T34429 C34IPU 155525488 EC50 < 30000 nM T34429 CK4PE0 155527401 IC50 = 21000 nM T34429 CFAY97 155528499 IC50 = 45300 nM T34429 CLYV89 155530137 Ki = 22.5 nM T34429 C9P0GH 155531194 IC50 = 611000 nM T34429 CHQC27 155532663 EC50 = 2100 nM T34429 C7AB8M 155532928 IC50 = 56000 nM T34429 C3VOB7 155532967 Ki = 62.3 nM T34429 CO07HD 155533348 Ki = 91.3 nM T34429 CB5FQ0 155533505 EC50 = 3540 nM T34429 CZ7Y6P 155536185 EC50 = 30000 nM T34429 CPXT08 155536463 EC50 = 3200 nM T34429 CY7M4G 155537329 EC50 = 2290 nM T34429 CMK0U4 155537399 Ki = 38.8 nM T34429 C84TLX 155537729 EC50 = 1270 nM T34429 C9JW6A 155537780 EC50 = 160 nM T34429 CI2Y1V 155539988 EC50 = 6450 nM T34429 C6FMK8 155541765 EC50 = 5400 nM T34429 C1S2TZ 155544028 IC50 = 353.6 nM T34429 CPO51I 155544666 EC50 = 7630 nM T34429 C79MRE 155546224 EC50 = 3190 nM T34429 C8U0GF 155546368 EC50 = 3340 nM T34429 C3DAN1 155546593 EC50 = 1190 nM T34429 CM50TS 155547626 Ki = 10.9 nM T34429 CD4HZ5 155548061 EC50 = 70 nM T34429 CDZ53Y 155548165 IC50 = 9590 nM T34429 CIDV89 155548253 EC50 = 4320 nM T34429 CI6NF7 155548271 EC50 = 69 nM T34429 C5ULB4 155550485 EC50 = 1600 nM T34429 CP1C6W 155550683 EC50 = 8500 nM T34429 CE07JY 155552244 EC50 = 5490 nM T34429 CROV92 155554398 Ki = 127 nM T34429 CM98WT 155555203 EC50 = 48 nM T34429 C8ZSP5 155555548 EC50 = 20417.38 nM T34429 CUJ1W6 155556119 IC50 = 63.1 nM T34429 CGQ5K1 155557728 EC50 = 920 nM T34429 C9H8YM 155558359 EC50 = 1970 nM T34429 CRA1Q8 155559251 EC50 = 3310 nM T34429 C5M9YR 155559414 EC50 = 690 nM T34429 C17ZAD 155560732 EC50 = 4570 nM T34429 C9KR3W 155560936 EC50 = 120 nM T34429 C07JNC 155562264 EC50 = 24 nM T34429 CN1R5L 155563200 EC50 > 13300 nM T34429 CL79NV 155563990 IC50 > 10000 nM T34429 C6Z1EK 155565097 EC50 = 890 nM T34429 CMO95H 155565655 EC50 < 30000 nM T34429 CUG7K4 155565793 EC50 = 530 nM T34429 CL90AG 155566198 EC50 = 230 nM T34429 CEMY87 155567089 EC50 = 1800 nM T34429 C04DGH 155567650 EC50 = 360 nM T34429 CR24FZ 155568280 Ki = 66800 nM T34429 CG4N5J 11515460 EC50 = 25.12 nM T34429 CB0LH8 11602721 EC50 = 7.943 nM T34429 C0V4ZT 11610777 EC50 = 31.62 nM T34429 CK74XW 11610796 EC50 = 25.12 nM T34429 CTAK49 11660066 EC50 = 7.943 nM T34429 CEG1P8 11688171 EC50 = 15.85 nM T34429 C7NWZ6 442202 IC50 = 13800 nM T34429 CDE0U8 44564586 EC50 = 630.96 nM T34429 C5V4IE 44564587 EC50 = 1258.93 nM T34429 C7UF0W 44564588 EC50 = 630.96 nM T34429 CUZ1D8 44564663 EC50 = 7.943 nM T34429 C0DHL2 44565105 EC50 = 1258.93 nM T34429 CAK86M 44565106 EC50 = 7943.28 nM T34429 C3X1FK 44565107 EC50 = 794.33 nM T34429 C2M1JA 44565108 EC50 = 1995.26 nM T34429 CG4BD2 44565109 EC50 = 1258.93 nM T34429 CFO01W 44565110 EC50 = 1258.93 nM T34429 COFX65 44565153 EC50 = 1000 nM T34429 C54KNB 44565154 EC50 = 1000 nM T34429 C6R1HF 44565155 EC50 = 630.96 nM T34429 CIFJ65 44565156 EC50 = 630.96 nM T34429 CF3OR4 44565157 EC50 = 316.23 nM T34429 CX5JK9 44565158 EC50 = 316.23 nM T34429 CL2DE7 44565207 EC50 = 1258.93 nM T34429 C0B1PF 44565208 EC50 = 316.23 nM T34429 CC25NX 44565209 EC50 = 125.89 nM T34429 CC1E2Z 71201944 EC50 = 1600 nM T34429 D00EJS 16054 EC50 = 1000000 nM T34429 D01SHB 3845 IC50 = 7000 nM T34429 D02LWF 44274422 IC50 = 1.1 nM T34429 D03FPQ 311434 EC50 = 158.49 nM T34429 D03JPN 11173546 Ki = 17 nM T34429 D06FLU 10480509 Ki = 95000 nM T34429 D07ZZD 9794818 Ki = 22.5 nM T34429 D08HTF 44240744 EC50 = 4200 nM T34429 D09BSE 10409038 Ki = 83000 nM T34429 D0C9TY 16727408 Ki = 2 nM T34429 D0D4LF 310378 EC50 = 3400 nM T34429 D0DA1E 23642319 EC50 = 212 nM T34429 D0IP9V 10107234 Ki = 9 nM T34429 D0LH4L 10154 Ki = 67000 nM T34429 D0O5EZ 854023 Ki = 22 nM T34429 D0R4RN 1204 Ki = 2.7 nM T34429 D0T9SK 6380 Ki = 2300 nM T34429 D0UH8F 44274190 IC50 = 8 nM T34429 D0V0AW 9823180 Ki = 71000 nM T34429 D0V2KB 44423690 Ki = 21000 nM T34429 D0X7CX 31762 Ki = 10500 nM T34429 D0X7HD 11184481 Ki = 16.4 nM T64765 D00JVR 2267 Ki = 147.91 nM T64765 D01AXB 60835 Ki > 5000 nM T64765 D01UTL 2995 Ki > 5000 nM T64765 D01ZII 2726 Ki > 1000 nM T64765 D03KQF 4011 Ki > 1000 nM T64765 D04USC 774 EC50 = 2.512 nM T64765 D05QNO 2968 IC50 = 820 nM T64765 D0AN7B 896 Ki = 0.5 nM T64765 D0B0CP 667467 Ki > 1000 nM T64765 D0NS6H 3152 IC50 = 350 nM T64765 D0P5SA 3372 Ki > 1000 nM T64765 D0TR5X 3386 Ki = 7300 nM T64765 D0Y5UG 2160 Ki > 1000 nM T64765 D0Z1RV 135398737 Ki = 631 nM T64765 D01UUD 9948102 Ki = 0.16 nM T64765 D02DTQ 24745335 Ki = 186.21 nM T64765 D04LSD 9818903 Ki = 0.4 nM T64765 D07YGH 9976892 Ki = 0.1 nM T64765 D0A3CL 49801838 IC50 = 400 nM T64765 D0EQ9T 24771368 Ki = 1.4 nM T64765 D0LI1C 44469321 IC50 > 10000 nM T64765 D0M4UZ 24994634 Ki = 1043 nM T64765 D0M8OC 16061509 Ki = 5.4 nM T64765 D0M9RQ 11697697 Ki = 0.5312 nM T64765 D0N8QK 24743471 Ki = 1.9 nM T64765 D0OW9L 11973780 IC50 = 0.33 nM T64765 D0R2OU 25070031 EC50 = 1.1 nM T64765 D02KAF 10103168 EC50 = 57.54 nM T64765 D05FYA 3035905 Ki = 6.5 nM T64765 D0B4TT 17747460 Ki = 0.2512 nM T64765 D0Q5YF 6450823 Ki = 2.138 nM T64765 C5H9CN 9287 Ki > 10000 nM T64765 C6C2BM 29296 Ki = 47.86 nM T64765 C2VQH8 29298 Ki = 9.7 nM T64765 CXH45A 170389 EC50 = 39.81 nM T64765 C2VRP9 182527 EC50 = 7.586 nM T64765 CUO7A3 203096 Ki > 501.19 nM T64765 CT7G3F 550705 IC50 = 11 nM T64765 CX0ZJ3 565544 EC50 = 0.123 nM T64765 CC72JQ 594090 Ki = 162.18 nM T64765 CXHE03 847672 Ki = 22 nM T64765 C89DBR 1072350 Ki = 600 nM T64765 CO8I4S 1203569 Ki = 1230 nM T64765 C42UIY 1394282 Ki = 4466.84 nM T64765 C5M1NP 2057716 Ki = 255 nM T64765 CK7RQ3 2057752 Ki = 22 nM T64765 C2SAZ9 2057757 Ki = 53.5 nM T64765 CCUB82 2057867 Ki = 265 nM T64765 CT8KN9 2232766 Ki = 53.9 nM T64765 CHQ4A3 2237924 Ki = 61.8 nM T64765 CUG96B 2238059 Ki = 52.9 nM T64765 C3WTG8 2843471 Ki = 427 nM T64765 C9J8KM 2922263 Ki = 140 nM T64765 C2XF9R 3002005 IC50 = 0.6 nM T64765 CAM7I6 3041343 Ki = 562.34 nM T64765 CL3BA9 3201696 IC50 = 900 nM T64765 CE0OK2 3209694 IC50 = 285 nM T64765 CM76PK 3209702 IC50 = 31 nM T64765 C1JU8E 3939214 EC50 = 3162.28 nM T64765 CQ43KY 4563101 Ki = 5011.87 nM T64765 CI5VZ7 6433105 Ki = 2.138 nM T64765 CRY54T 8434659 Ki = 114.5 nM T64765 CM95CG 9119245 IC50 = 1370 nM T64765 C4V5IX 9793791 EC50 = 19.5 nM T64765 C24GNE 9798145 Ki = 0.5012 nM T64765 C5ON0J 9798429 Ki = 1.2 nM T64765 C5Z2KM 9805944 Ki = 9.3 nM T64765 CW3A8U 9814674 Ki = 0.5012 nM T64765 C74RIY 9816601 Ki = 19.05 nM T64765 CIH80R 9818650 Ki = 1.738 nM T64765 C37YHS 9834709 Ki = 107.15 nM T64765 CHFI61 9835304 Ki = 0.9333 nM T64765 C2XA5B 9835305 Ki = 3 nM T64765 C2YJF1 9836681 Ki = 1.479 nM T64765 CBPZ27 9836953 Ki = 5.495 nM T64765 C03JZN 9838864 Ki = 1.6 nM T64765 C9WZL0 9839643 Ki = 13 nM T64765 CO0L4B 9840607 Ki = 0.8 nM T64765 CKNF95 9840856 Ki = 0.75 nM T64765 C2MR5U 9841261 Ki = 2 nM T64765 CT5M1L 9851785 Ki = 15 nM T64765 CZB9K7 9858195 Ki = 2.1 nM T64765 C3I4PF 9858858 Ki = 0.2188 nM T64765 CDQ91J 9862335 Ki = 1.9 nM T64765 CB4W3Z 9865378 Ki = 4 nM T64765 CB7RF9 9866657 Ki = 26 nM T64765 C97BPS 9873094 Ki = 1.585 nM T64765 CX63EL 9878125 Ki = 28.18 nM T64765 CPF15V 9878707 Ki = 3.02 nM T64765 C3O5JL 9879041 Ki = 1.622 nM T64765 C2VN5R 9879473 Ki = 1.95 nM T64765 C2G7ZL 9880039 Ki = 0.871 nM T64765 C34AHG 9880208 Ki = 8.318 nM T64765 C0G4RM 9880373 Ki = 2.239 nM T64765 CQ4PW7 9880608 Ki = 0.5129 nM T64765 C6A5OE 9880698 Ki = 1.413 nM T64765 CS9R4U 9883980 Ki = 0.95 nM T64765 C4ZMS0 9884637 Ki = 0.4 nM T64765 CO2RP1 9884652 Ki = 0.08 nM T64765 CF3A4Q 9899875 Ki = 66.07 nM T64765 C0E7WN 9901568 Ki = 2.291 nM T64765 CTG3J8 9902060 Ki = 1.698 nM T64765 CX40PG 9902719 Ki = 7.762 nM T64765 C5AX3I 9902971 Ki = 3 nM T64765 CYWQ50 9906447 Ki = 0.2692 nM T64765 C8H0OF 9921577 Ki = 12.88 nM T64765 CWQ75J 9923147 Ki = 6.166 nM T64765 CZ02FE 9923162 EC50 = 1584.89 nM T64765 CI3V0F 9923186 Ki = 19.5 nM T64765 CT70EV 9923762 Ki = 13 nM T64765 C3QCB0 9925192 Ki = 11 nM T64765 CKIF45 9925337 Ki = 0.2042 nM T64765 CV9QC1 9926445 Ki = 8.913 nM T64765 CX5GL1 9928224 Ki = 1.7 nM T64765 CFKT60 9943711 Ki = 32.36 nM T64765 CEZ12V 9944320 Ki = 1.23 nM T64765 CA0B8C 9944610 Ki = 0.8 nM T64765 CX8O7C 9945134 Ki = 8.318 nM T64765 CKH0S9 9945319 Ki = 10 nM T64765 CBT83O 9945660 Ki = 5 nM T64765 CW9TE0 9946163 Ki = 22 nM T64765 CJ83MW 9946194 Ki = 1 nM T64765 CVN18W 9946461 Ki = 0.1 nM T64765 CKQ28I 9947227 Ki = 1.698 nM T64765 CBIP87 9947283 Ki = 43 nM T64765 C8J0UF 9951524 Ki = 0.54 nM T64765 C8J9FY 9951566 Ki = 1 nM T64765 CQ9LU7 9951970 Ki = 74 nM T64765 CJ7GM8 9953505 Ki = 16 nM T64765 CCO8U5 9954017 Ki = 0.4074 nM T64765 CL56QZ 9957437 Ki = 6633 nM T64765 CP9I3U 9964223 Ki = 141.25 nM T64765 C7JV1Y 9965041 Ki = 15.14 nM T64765 C74TEM 9966707 Ki = 0.631 nM T64765 C1PMY8 9967362 Ki = 1.349 nM T64765 C9DY6F 9967363 Ki = 13.49 nM T64765 CF36IJ 9968975 Ki = 19 nM T64765 CXU79I 9969015 Ki = 6 nM T64765 CP1W9B 9969328 Ki = 0.08511 nM T64765 CCO7G5 9971374 Ki = 3.981 nM T64765 C8UE9A 9972181 Ki = 10 nM T64765 C1IZP8 9973087 Ki = 0.26 nM T64765 CC57WG 9973932 Ki = 0.2 nM T64765 C07LHX 9974962 Ki = 54 nM T64765 C17UZA 9977652 Ki = 0.5012 nM T64765 CA2E5N 9994551 Ki = 3.162 nM T64765 CA6JE9 9995111 Ki = 156 nM T64765 C8VRW9 9997377 Ki = 0.12 nM T64765 C5F6HZ 9999254 Ki = 141 nM T64765 CB36IL 10000114 Ki = 0.53 nM T64765 CJG5P8 10003715 Ki = 1.2 nM T64765 CP4F7M 10015825 Ki = 52 nM T64765 C1H9RS 10017117 Ki = 100 nM T64765 CUN7T8 10019811 Ki = 0.16 nM T64765 CZ7QH8 10021441 Ki = 0.2512 nM T64765 CIF8E2 10023270 Ki = 6 nM T64765 CPGA98 10023327 Ki = 1.047 nM T64765 C1L5DN 10026806 Ki = 18 nM T64765 C25DHA 10037650 Ki = 6309.57 nM T64765 C32SGR 10041484 Ki = 19.95 nM T64765 C1WH8Q 10042344 Ki = 2.5 nM T64765 CXDZ96 10042900 Ki = 0.2399 nM T64765 CB9EF4 10044556 Ki = 27.3 nM T64765 C9DQ3G 10045080 Ki = 0.1585 nM T64765 CJ5R2I 10045991 Ki = 0.3162 nM T64765 CIZ35V 10048448 Ki = 17 nM T64765 C8Y6NF 10063514 Ki > 300 nM T64765 C12XIY 10063835 Ki = 194 nM T64765 CMUW84 10064805 Ki = 6.607 nM T64765 CK38NM 10065106 Ki = 0.7943 nM T64765 CB2OY4 10066872 Ki = 0.4365 nM T64765 CLN7P8 10067030 Ki = 48.98 nM T64765 C0ARK3 10067161 Ki = 0.091 nM T64765 CU78GI 10067368 Ki = 10 nM T64765 CV0PL3 10067493 Ki = 2.9 nM T64765 C76MHL 10070496 Ki = 1 nM T64765 C3R6NL 10085528 Ki = 19.95 nM T64765 C76PGV 10086941 Ki = 600 nM T64765 CRC0G2 10087134 Ki = 4.2 nM T64765 CMKD76 10087533 Ki = 10 nM T64765 C8G1PU 10087576 Ki = 0.4 nM T64765 C2JAM3 10088337 Ki = 10 nM T64765 CO9RH2 10088634 Ki = 0.1778 nM T64765 CH14BN 10089061 Ki = 0.3 nM T64765 CE4I5T 10090759 Ki = 17.1 nM T64765 CRBM02 10090854 Ki = 41 nM T64765 CB12MS 10093180 Ki = 1 nM T64765 C9LG7V 10093599 Ki = 6.166 nM T64765 CB0P7C 10106063 Ki = 1995.26 nM T64765 C0MWB3 10106318 Ki = 14 nM T64765 CYQ71B 10107667 Ki = 25 nM T64765 CGC06P 10109296 Ki = 5 nM T64765 CVYQ41 10109322 Ki = 0.52 nM T64765 C0FO9Y 10109898 Ki = 0.26 nM T64765 C2F0WU 10110088 Ki = 0.52 nM T64765 CJW21B 10110274 Ki = 14 nM T64765 CI32TX 10111190 Ki = 1900 nM T64765 C37VXH 10114059 Ki = 37 nM T64765 CW91OK 10130526 Ki = 11 nM T64765 CATZ34 10131633 Ki = 0.7413 nM T64765 C6L5QN 10131681 Ki = 0.5888 nM T64765 C7LUR3 10131721 Ki = 1.148 nM T64765 C5JHK9 10132217 Ki = 7 nM T64765 CPK34U 10132440 Ki = 0.21 nM T64765 CFL03W 10132505 Ki = 16 nM T64765 CZOH16 10132506 Ki = 40 nM T64765 CG2RN3 10133403 Ki = 0.8318 nM T64765 CVC16Q 10133949 Ki = 0.2042 nM T64765 CP64RT 10134089 Ki = 3 nM T64765 CJMW34 10136423 Ki = 500 nM T64765 CI4SB1 10149516 Ki = 0.6761 nM T64765 C3NEB7 10149527 Ki = 1.096 nM T64765 CLQV76 10149817 Ki = 5.248 nM T64765 CD78PH 10154945 Ki = 0.51 nM T64765 C68VZN 10155386 Ki = 3 nM T64765 CC43NE 10155398 Ki = 0.955 nM T64765 CKBI53 10156476 Ki = 2 nM T64765 C28DJV 10156706 Ki = 0.35 nM T64765 C9Z8FG 10172984 Ki = 3.467 nM T64765 CTZ6D4 10176370 EC50 = 12.59 nM T64765 CIY6O1 10177442 Ki = 2.042 nM T64765 C1BOA5 10177656 Ki = 6 nM T64765 CG9VU3 10177769 Ki = 1300 nM T64765 C2PZF9 10177985 Ki = 15 nM T64765 CRAF12 10178641 Ki = 0.045 nM T64765 C6VJ4E 10178836 Ki = 1500 nM T64765 CLU70K 10179531 Ki = 1.514 nM T64765 C1BDR3 10179589 Ki = 870 nM T64765 C7EAS8 10179744 Ki = 4 nM T64765 CMY04N 10193075 Ki = 0.6166 nM T64765 CA2JV0 10193212 Ki = 0.5129 nM T64765 CF78GC 10193234 Ki = 1.738 nM T64765 CB7VM4 10193648 Ki = 0.7586 nM T64765 CDM8J7 10197870 EC50 = 39.81 nM T64765 CJ19SV 10200160 Ki = 4 nM T64765 CEC9S3 10200613 Ki = 1100 nM T64765 CL1SW8 10200614 Ki = 1.995 nM T64765 C5SFB4 10201558 Ki = 4 nM T64765 CMY9U5 10202400 Ki = 7900 nM T64765 C2HE9F 10214918 Ki = 1.349 nM T64765 CEZ9F3 10215178 Ki = 0.9772 nM T64765 CI8A0S 10215179 Ki = 0.7244 nM T64765 CU1KG6 10223051 Ki = 1.445 nM T64765 C1KRJ3 10226345 Ki = 2900 nM T64765 CA1H7G 10236303 Ki = 0.912 nM T64765 CS8GC6 10236461 Ki = 81.28 nM T64765 CQH8W7 10236617 Ki = 5.012 nM T64765 CC2MH8 10243990 Ki = 29 nM T64765 CN4G5C 10244716 Ki = 0.2512 nM T64765 C71OKT 10246785 Ki = 1.549 nM T64765 CWE2N8 10247391 Ki = 0.1995 nM T64765 C74IWR 10247831 Ki = 0.81 nM T64765 CFZQ39 10249083 Ki = 0.7943 nM T64765 C6N1IJ 10261471 Ki = 10 nM T64765 CHLG27 10266140 Ki = 2.512 nM T64765 CX6F1A 10267432 Ki = 129 nM T64765 C8R9AO 10268635 Ki = 6 nM T64765 CS6MU7 10268636 Ki = 8.511 nM T64765 C3DMT5 10269256 Ki = 46 nM T64765 C96ZXH 10269924 IC50 = 0.98 nM T64765 C9D2QB 10270093 Ki = 2 nM T64765 CXQY92 10270155 Ki = 0.43 nM T64765 CXH54Q 10270357 Ki = 0.19 nM T64765 C4VJ8Z 10286408 Ki = 0.7762 nM T64765 C4HT5F 10286561 Ki = 0.8913 nM T64765 C8ED3N 10286858 Ki = 0.5495 nM T64765 CC02JT 10291205 Ki = 15 nM T64765 C1U4CD 10291260 Ki = 1 nM T64765 C73ESP 10291489 Ki = 2 nM T64765 CH39FK 10292436 Ki = 0.19 nM T64765 C5DQ4K 10292893 Ki = 5 nM T64765 CN9HR1 10294844 Ki = 1.995 nM T64765 CCXD16 10295613 Ki = 3 nM T64765 CBNQ58 10308670 Ki = 3.802 nM T64765 CP10NL 10314462 Ki = 2.089 nM T64765 CL8XC6 10319869 Ki = 2.291 nM T64765 C8IU6A 10320608 Ki = 2.2 nM T64765 CLKX29 10335984 Ki = 0.76 nM T64765 CCI2F5 10339638 Ki = 0.2 nM T64765 C7ENH1 10339677 Ki = 0.1585 nM T64765 CMY17D 10358078 Ki > 300 nM T64765 CIYQ04 10358984 Ki = 3.8 nM T64765 CGRE95 10359169 Ki = 0.84 nM T64765 CGQN51 10359235 Ki = 0.8 nM T64765 C2QJX3 10360149 Ki = 5.8 nM T64765 C4OJ2X 10360264 Ki = 2.2 nM T64765 CGT03L 10360801 Ki = 8.61 nM T64765 CR5V4N 10360920 Ki = 2.884 nM T64765 CZ1V6E 10361356 Ki = 0.07943 nM T64765 CRW81V 10362005 Ki = 42.3 nM T64765 CM31KG 10364005 Ki = 31 nM T64765 C8FP3M 10364480 Ki = 7.3 nM T64765 CB3PD0 10364831 Ki = 44.67 nM T64765 CY14NQ 10365527 Ki = 3.467 nM T64765 CI2C4X 10381075 Ki = 0.34 nM T64765 C8OCF0 10381995 Ki = 11.6 nM T64765 CBO49T 10382001 Ki = 0.72 nM T64765 CL18SQ 10382998 Ki = 17.78 nM T64765 CS8EO3 10384556 Ki = 187 nM T64765 CL8O4S 10387446 Ki > 300 nM T64765 CF7KV2 10399784 Ki = 100 nM T64765 C76WZF 10401439 Ki = 7.4 nM T64765 CV3Q4J 10406178 Ki = 15.85 nM T64765 C84DJP 10408272 Ki = 0.1995 nM T64765 C7GJE9 10419556 EC50 = 794.33 nM T64765 CHD8X9 10423494 Ki = 158.49 nM T64765 C6RVC0 10426237 Ki = 0.7943 nM T64765 C6GXW2 10426299 Ki = 2.5 nM T64765 CWV8M6 10426540 Ki = 0.4898 nM T64765 CRD8H9 10427511 Ki = 4.571 nM T64765 C6KR8Z 10428027 Ki = 0.19 nM T64765 C4NJ7H 10428707 Ki = 5 nM T64765 C1G6TW 10428924 Ki = 0.5012 nM T64765 CE8N2K 10429016 Ki = 7.943 nM T64765 CI0LK6 10429386 Ki = 0.5012 nM T64765 CA6PK0 10430564 Ki = 0.3162 nM T64765 CE15WN 10446240 IC50 = 1.259 nM T64765 C80TCL 10450279 Ki = 0.36 nM T64765 C2NP4V 10451051 Ki = 2.399 nM T64765 CMC6S4 10451557 Ki = 12.1 nM T64765 CKOB53 10452164 Ki = 0.38 nM T64765 CWJ41L 10452501 Ki = 273 nM T64765 CQ6B1C 10452629 Ki = 22.6 nM T64765 CP76CB 10452850 Ki = 1 nM T64765 CA4Z8J 10468601 Ki = 7.943 nM T64765 C0PTH3 10470098 Ki = 2.63 nM T64765 CKVN59 10471844 Ki = 8.71 nM T64765 CRM27I 10472082 Ki = 0.6761 nM T64765 CI7D9Z 10473209 Ki = 0.1905 nM T64765 COG21I 10473695 Ki = 0.5012 nM T64765 CTU89N 10477013 Ki = 5.888 nM T64765 CK8NO7 10515050 Ki = 8.3 nM T64765 C6O1ZI 10515993 Ki = 41 nM T64765 CZM34W 10537958 Ki = 15 nM T64765 CS35LU 10538833 Ki = 42 nM T64765 CGW14S 10545988 Ki = 141.25 nM T64765 C0MVL8 10548835 Ki = 75 nM T64765 C6SGD5 10583206 EC50 = 776.25 nM T64765 CX6G7H 10591811 Ki = 118 nM T64765 C6L4YF 10660486 Ki = 91 nM T64765 CBMH01 10678418 Ki = 870.96 nM T64765 CR8WH9 10678661 EC50 = 100 nM T64765 CH5N3M 10680963 Ki = 42 nM T64765 C9O3AL 10688021 Ki = 8.3 nM T64765 CD7I4S 10702196 Ki = 11481.54 nM T64765 C4DKQ5 10715823 Ki = 37 nM T64765 CWR1T8 10715857 Ki = 41 nM T64765 C56JNC 10760516 Ki = 169.82 nM T64765 CTG0S1 10773349 EC50 = 269.15 nM T64765 CE8ZO0 10776393 Ki = 4.7 nM T64765 CF6D2A 10777275 Ki = 19 nM T64765 C16RQB 10800875 Ki = 13 nM T64765 C03SWA 10820929 Ki = 2511.89 nM T64765 CDI46B 10820930 Ki = 19952.62 nM T64765 CY89MD 10861302 Ki = 9.9 nM T64765 CI06PY 10870282 Ki = 123 nM T64765 C5XL0G 10873565 Ki = 0.5012 nM T64765 CTC3W5 10879463 Ki = 18620.87 nM T64765 C3PSF4 10879621 Ki = 6.7 nM T64765 C0K9EH 10882243 Ki = 92 nM T64765 CR86MN 10902522 Ki = 77 nM T64765 CQ0UK9 10902577 Ki = 1130 nM T64765 CX1M6V 10903015 Ki = 119 nM T64765 CWR49U 10904105 Ki = 18 nM T64765 C6ZEQ5 10904475 Ki = 114 nM T64765 CJC05L 10913722 Ki = 378 nM T64765 CB5V2T 10916261 Ki = 0.07943 nM T64765 C3A7KJ 10926938 Ki = 157 nM T64765 C7BS3K 10933521 Ki = 20 nM T64765 CYA27N 10934158 EC50 = 190.55 nM T64765 C4GUE5 10935978 Ki = 124 nM T64765 CR8F3C 10936212 Ki = 84 nM T64765 CX37ZO 10945113 EC50 = 9549.93 nM T64765 C0LPS6 10947603 Ki = 95 nM T64765 CMZ1E9 10947780 Ki = 88 nM T64765 COC26R 10948079 Ki = 201 nM T64765 CSBX68 10949464 Ki = 0.75 nM T64765 C3IBD5 10956157 Ki = 191 nM T64765 CN82HV 10956568 Ki = 362 nM T64765 C5NVO7 10956869 Ki = 9.7 nM T64765 CWGK20 10957911 Ki = 7.6 nM T64765 CEK4O6 10958276 Ki = 253 nM T64765 CWU67L 10959016 Ki = 125 nM T64765 CBL8S0 10969785 Ki = 50 nM T64765 C0ZT6K 10977121 Ki = 5.4 nM T64765 CI63DO 10977922 Ki = 6 nM T64765 CA95TC 10978141 EC50 = 91.2 nM T64765 CCM7X8 10978306 Ki = 8.2 nM T64765 C1D5SW 10978949 Ki = 411 nM T64765 CB4E5X 10978950 Ki = 90 nM T64765 C4QV2F 10979638 Ki = 1.23 nM T64765 CV9W8X 10980245 Ki = 34 nM T64765 C4J5UT 10980927 Ki = 27 nM T64765 CF15CY 10986211 EC50 = 2330 nM T64765 CA59XG 10990520 Ki = 149 nM T64765 CY0J2X 10993098 Ki = 12 nM T64765 C9S8MQ 11003651 Ki = 0.5012 nM T64765 CHLQ20 11004759 Ki = 0.3162 nM T64765 CM4O2L 11012518 Ki = 50.12 nM T64765 C21FJM 11012519 Ki = 630.96 nM T64765 C4JI8P 11014530 Ki = 90 nM T64765 C8CK1J 11021932 Ki = 85 nM T64765 CEG0C2 11023683 Ki = 87 nM T64765 C0RMP8 11023756 Ki = 257 nM T64765 CZ2QO9 11025405 Ki = 761 nM T64765 C26GSM 11025896 Ki = 107 nM T64765 CZI50D 11033823 Ki = 15 nM T64765 CH1E9J 11034870 Ki = 42 nM T64765 C8WZT4 11035490 Ki = 167 nM T64765 CM10FQ 11036235 Ki = 2.8 nM T64765 C20DCR 11043445 Ki = 6309.57 nM T64765 CD4P6B 11044642 Ki = 126 nM T64765 C1JV6N 11045549 Ki = 78 nM T64765 C51KER 11048988 Ki = 1.995 nM T64765 CK4Z3A 11066841 Ki = 163 nM T64765 CZTL25 11067710 Ki = 169 nM T64765 C83AJC 11078658 Ki = 1130 nM T64765 C54LKV 11080253 Ki = 1.5 nM T64765 CAZ0H8 11086114 Ki = 7943.28 nM T64765 CVO58P 11091279 Ki = 32 nM T64765 CO81WF 11094685 EC50 > 0.0001 nM T64765 C71OCL 11107010 Ki = 119 nM T64765 CWQ06X 11110358 Ki = 26 nM T64765 C5GXC9 11111856 Ki = 550 nM T64765 CWE5L2 11116130 EC50 > 0.0001 nM T64765 C3WSQ0 11122095 Ki = 1.8 nM T64765 C2LC7H 11122254 Ki = 238 nM T64765 CUF10O 11126319 EC50 = 96 nM T64765 CNA91S 11129149 Ki = 32 nM T64765 C6VEC5 11130677 Ki = 19 nM T64765 C7O4LG 11131540 Ki = 37 nM T64765 CU5H7C 11148240 Ki = 93.33 nM T64765 CU9DJ0 11159854 Ki = 83.18 nM T64765 CXI5N2 11163942 Ki = 0.62 nM T64765 C6CY2H 11164099 EC50 = 3.981 nM T64765 CQ0T9Y 11166138 Ki = 158.49 nM T64765 CON91C 11171320 Ki = 181.97 nM T64765 CP1KD2 11174563 Ki = 0.9 nM T64765 CR3XM0 11175719 Ki = 8.5 nM T64765 CX0I3V 11178286 EC50 = 31.62 nM T64765 C75PYH 11187623 Ki = 0.2455 nM T64765 C0WJ6I 11189201 EC50 = 79.43 nM T64765 C1KUT6 11200224 Ki = 2100 nM T64765 CSF2E5 11206058 Ki = 1174.9 nM T64765 C8TI6J 11210869 EC50 = 7.943 nM T64765 CT28FP 11219164 Ki = 758.58 nM T64765 CK5UX6 11223503 Ki = 31.62 nM T64765 CW0UH1 11232370 Ki = 0.96 nM T64765 CXTC95 11232950 Ki = 0.4898 nM T64765 C3Z0JI 11234485 Ki = 1.4 nM T64765 CT4UQ6 11234833 Ki = 300 nM T64765 CMW61C 11235785 Ki = 79.43 nM T64765 C6Q8IR 11240759 EC50 = 6.761 nM T64765 C2VU5G 11241109 Ki > 10000 nM T64765 CL81BT 11244101 Ki = 3.4 nM T64765 CA1XB4 11249610 Ki = 4.8 nM T64765 CJ4E3B 11252330 EC50 = 2754.23 nM T64765 CCH3M5 11255988 Ki = 0.69 nM T64765 CE5J6L 11256632 Ki = 4.8 nM T64765 CV47MB 11257330 Ki = 110 nM T64765 CJ83BQ 11266328 Ki = 5370.32 nM T64765 CD3UV9 11275349 EC50 = 2.344 nM T64765 CAZX95 11279886 Ki = 24 nM T64765 C5LNK1 11283135 Ki = 0.871 nM T64765 CSX09V 11286909 EC50 = 912.01 nM T64765 CRO65G 11290442 Ki = 0.2692 nM T64765 CA5UI2 11291550 Ki = 63.1 nM T64765 CD02TP 11302722 Ki = 3 nM T64765 CI5XH2 11303905 Ki = 1.1 nM T64765 CJS9C0 11304851 IC50 > 3200 nM T64765 C9L0IK 11313056 Ki = 0.89 nM T64765 CYL61U 11327520 EC50 = 15.85 nM T64765 CG8TW1 11328347 Ki = 110 nM T64765 C9SKQ1 11336447 Ki = 0.74 nM T64765 C9IB0R 11336692 EC50 = 2.512 nM T64765 C6OAT4 11337639 Ki = 63.1 nM T64765 CR37ZU 11340988 Ki = 0.4365 nM T64765 C3HE1G 11344458 EC50 = 30.9 nM T64765 C3JW0L 11349657 Ki = 2 nM T64765 CC13FL 11349921 Ki = 1.8 nM T64765 CYG18L 11368217 Ki = 81.28 nM T64765 CO2X1F 11371282 Ki = 2.3 nM T64765 C28TIF 11371853 Ki = 323 nM T64765 C6JCT1 11374202 Ki = 39.81 nM T64765 C5ZHK8 11393516 Ki = 8.318 nM T64765 CV3E2R 11394346 Ki = 0.2291 nM T64765 CW16YE 11395725 EC50 = 3.981 nM T64765 C4YZM0 11407784 EC50 = 7.943 nM T64765 CTP83F 11412714 Ki = 2818.38 nM T64765 CZXC10 11416895 EC50 = 25.12 nM T64765 CP8D1E 11418968 EC50 = 15.85 nM T64765 CG4P9O 11440060 Ki > 1000 nM T64765 CF0LA9 11440968 Ki = 2.7 nM T64765 CD29ST 11450972 Ki = 0.871 nM T64765 C36YEK 11458595 Ki = 4265.8 nM T64765 CPI63U 11461249 Ki = 24 nM T64765 CW86EQ 11461930 Ki = 18 nM T64765 C3B1LH 11469514 Ki = 15.49 nM T64765 C6E3CJ 11473403 Ki = 93 nM T64765 C91NEG 11474535 Ki = 100 nM T64765 CI0WR7 11475310 Ki = 33 nM T64765 CL4W8O 11486222 Ki = 52 nM T64765 C7R3SY 11492189 Ki = 63.1 nM T64765 CH28CN 11495137 Ki = 2 nM T64765 CD4S0X 11499376 Ki = 630.96 nM T64765 CG9Z3H 11499453 Ki = 1.585 nM T64765 CFO2Z5 11499454 Ki = 39.81 nM T64765 CMO8P5 11500302 Ki = 4.467 nM T64765 C9K2VE 11501382 Ki = 0.34 nM T64765 CWK6Z7 11501506 Ki = 4 nM T64765 C6HM0U 11501983 IC50 = 1.5 nM T64765 CI62OX 11502343 Ki = 0.1562 nM T64765 CPO8S1 11502381 Ki = 0.07812 nM T64765 CGB8M5 11502401 Ki = 1.7 nM T64765 C2TVA0 11502638 Ki = 0.09375 nM T64765 CPUV18 11503379 Ki = 3 nM T64765 C1RQO0 11503600 Ki = 40 nM T64765 CVQR26 11506928 Ki = 39.81 nM T64765 CQ91UB 11507778 IC50 = 5 nM T64765 CH8O5U 11507838 Ki = 85 nM T64765 CRFV19 11508245 Ki = 23 nM T64765 C7QZX4 11508633 Ki = 62 nM T64765 C2URB1 11508788 Ki = 1.04 nM T64765 CZ61OG 11509486 Ki = 3.8 nM T64765 CA64UW 11509682 IC50 = 28 nM T64765 CDM01C 11510623 EC50 = 7 nM T64765 C96WEL 11515374 Ki = 3.2 nM T64765 CO0T6Q 11516310 Ki = 0.4 nM T64765 C17QPU 11516322 Ki = 0.34 nM T64765 CS24AX 11516386 Ki = 0.375 nM T64765 CNM42D 11516387 Ki = 0.5 nM T64765 C6X1AJ 11516392 Ki = 0.1 nM T64765 C5MSI4 11517190 Ki = 2 nM T64765 C20FMG 11517340 Ki = 0.1562 nM T64765 CPQN50 11517341 Ki = 0.1562 nM T64765 CG51XI 11518064 Ki = 9.3 nM T64765 CN30CY 11521414 Ki = 31.62 nM T64765 CHV83Z 11522780 Ki = 1.1 nM T64765 C5F0GK 11522882 Ki = 0.29 nM T64765 CM09RF 11524148 Ki = 1 nM T64765 CL09JW 11524225 Ki = 0.03125 nM T64765 CE4DK8 11530172 Ki = 679 nM T64765 C9CM4J 11530812 EC50 = 44 nM T64765 CV9X1J 11531102 IC50 = 45 nM T64765 CP1WJ6 11531115 Ki = 0.13 nM T64765 CJ89VE 11531261 IC50 = 23 nM T64765 CI6B3Q 11531262 Ki = 0.1259 nM T64765 CZ93HX 11531536 Ki = 0.89 nM T64765 C94AGK 11531634 Ki = 0.1 nM T64765 CZP0R5 11532060 Ki = 0.74 nM T64765 CS7Q6G 11532065 Ki = 0.1 nM T64765 CDX19H 11532153 Ki = 20 nM T64765 CKI40W 11533362 Ki = 0.3162 nM T64765 CL8SY6 11536119 Ki = 3.162 nM T64765 CT3EK1 11537851 IC50 = 49 nM T64765 C7R3HN 11538251 Ki = 0.2399 nM T64765 CST25V 11538747 IC50 = 21 nM T64765 C8GZ1I 11539020 Ki = 0.09375 nM T64765 CBMY10 11539128 Ki = 0.71 nM T64765 CIR9M2 11539598 Ki = 1.8 nM T64765 CI4RN5 11539608 Ki = 9.7 nM T64765 C32SDT 11540601 Ki = 2840 nM T64765 C1LNB3 11540902 Ki = 2 nM T64765 CEUW20 11544316 Ki = 0.31 nM T64765 CJYA71 11544339 Ki = 20 nM T64765 CC9HR6 11544498 Ki = 1.1 nM T64765 C5CO2F 11544608 Ki = 37 nM T64765 C9UG2V 11544758 Ki = 0.832 nM T64765 C19ZFG 11545034 Ki = 10 nM T64765 C4CDU5 11545613 IC50 = 91 nM T64765 CGE5W7 11546121 Ki = 0.34 nM T64765 CN0YI6 11546137 Ki = 1.22 nM T64765 CFNG56 11546387 Ki = 0.36 nM T64765 CQ53AN 11546625 Ki = 267 nM T64765 CE7L2Y 11551689 Ki = 27.6 nM T64765 C74HSR 11551775 Ki = 0.69 nM T64765 CVK67I 11551796 Ki = 5 nM T64765 CLA1Y8 11553091 EC50 = 9 nM T64765 CH0E4A 11553554 Ki = 1.7 nM T64765 CKT1O8 11554040 Ki = 0.1862 nM T64765 CMC79Y 11554762 Ki = 1.1 nM T64765 CKDY35 11557610 Ki = 3.981 nM T64765 CGO36J 11558917 Ki = 356 nM T64765 CC2NI5 11560214 IC50 = 11 nM T64765 CXQ5J6 11560724 Ki = 1.2 nM T64765 CL3C7W 11564628 Ki = 39.81 nM T64765 CBW07F 11566918 EC50 = 1 nM T64765 C92BED 11567158 Ki = 238 nM T64765 CZMB92 11567596 Ki = 0.2313 nM T64765 CP7W6H 11567952 Ki = 0.09375 nM T64765 C16AJG 11572015 Ki = 3.981 nM T64765 C3HB4N 11572939 Ki = 19.95 nM T64765 C2UL6M 11573592 Ki = 0.84 nM T64765 CP03BT 11573599 Ki = 110 nM T64765 C2DO3Z 11573764 Ki = 0.27 nM T64765 C5GCA9 11574091 Ki = 14 nM T64765 CCYD42 11574150 Ki = 0.22 nM T64765 CCKY21 11574624 Ki = 0.54 nM T64765 CM9G8H 11576666 Ki = 3 nM T64765 C49RMJ 11580790 Ki = 32 nM T64765 C7I5KM 11581252 Ki = 0.69 nM T64765 CE0U8J 11581337 Ki = 0.2188 nM T64765 C7MCE6 11581640 IC50 = 14 nM T64765 CZ28HJ 11581919 IC50 = 1.6 nM T64765 CICM46 11582059 Ki = 0.1 nM T64765 CZ1QI8 11582342 Ki = 2 nM T64765 C2J9NU 11582508 Ki = 7.4 nM T64765 C6D1MA 11584660 Ki > 316.23 nM T64765 CT4IW3 11587883 Ki = 4.4 nM T64765 CFSP59 11588013 Ki = 15 nM T64765 C6V1YG 11588680 Ki = 0.14 nM T64765 CO4X7S 11588992 Ki = 0.43 nM T64765 C5Q1VL 11590382 Ki = 106 nM T64765 CH49ZV 11595838 IC50 = 53 nM T64765 CI95MX 11595847 Ki = 0.31 nM T64765 COS24N 11596426 Ki = 0.4062 nM T64765 C46AUZ 11597035 Ki = 9.5 nM T64765 CN16CW 11600779 Ki = 7.943 nM T64765 CZ79UT 11600780 Ki = 79.43 nM T64765 CN7C5W 11600849 Ki = 5.012 nM T64765 CF7S2E 11602209 Ki = 54 nM T64765 C1GL6E 11602780 Ki = 4.7 nM T64765 C9THD4 11602952 Ki = 50 nM T64765 CP1S8M 11603022 Ki = 0.33 nM T64765 C9MK8D 11603156 EC50 = 54 nM T64765 C7T3WI 11603194 Ki = 2.9 nM T64765 C04ORX 11603648 Ki = 0.257 nM T64765 CKH76N 11603838 Ki = 2 nM T64765 CH32AR 11603948 Ki = 30 nM T64765 CMG3H1 11608543 Ki = 0.4467 nM T64765 CLS4E5 11609917 Ki = 5.8 nM T64765 C05MNI 11610190 Ki = 0.74 nM T64765 CD2PU0 11610816 IC50 = 1.6 nM T64765 CKXH63 11610910 Ki = 7 nM T64765 C5O4ND 11611851 IC50 = 3.6 nM T64765 CY4CA7 11615406 Ki = 39.81 nM T64765 C6NZ8Q 11615601 Ki = 15.85 nM T64765 CC5I0P 11616557 Ki = 12 nM T64765 CN5M3X 11617313 Ki = 119 nM T64765 C67KGT 11617839 Ki = 0.3 nM T64765 CD28IH 11618024 Ki = 0.06875 nM T64765 CZ4YP0 11618099 Ki = 87 nM T64765 C36OSA 11618702 Ki = 0.0625 nM T64765 C1F4DL 11618807 Ki = 6.5 nM T64765 C1GB6K 11618861 Ki = 0.4 nM T64765 CW0ZM6 11619260 EC50 = 2 nM T64765 CMC45P 11619374 Ki = 15 nM T64765 CUQ63N 11620342 Ki = 2606 nM T64765 CX2A1I 11622495 EC50 = 5.012 nM T64765 CG4HL6 11622672 Ki = 7.943 nM T64765 CB0O5X 11624178 Ki = 3.2 nM T64765 CNS92I 11624908 EC50 = 23 nM T64765 C7YMN1 11625318 Ki = 50 nM T64765 CKU1V9 11625356 IC50 = 387 nM T64765 CW5Z4A 11629829 Ki = 19.95 nM T64765 CP1E8B 11629931 Ki = 39.81 nM T64765 CS1D6C 11630921 Ki = 4.1 nM T64765 C6A2BH 11630954 Ki = 25.12 nM T64765 CYM9Q4 11631394 Ki = 12 nM T64765 CSA4K9 11631843 Ki = 0.4 nM T64765 C0G6PN 11632103 IC50 = 0.72 nM T64765 CE8PC0 11632364 Ki = 1.7 nM T64765 C9HCM6 11632711 Ki = 1.1 nM T64765 C7H0AV 11633028 Ki = 0.35 nM T64765 CK4M2L 11633374 Ki = 14 nM T64765 COB0P4 11634166 Ki = 28 nM T64765 C2PGB7 11637064 Ki = 31.62 nM T64765 C9LS8Y 11638162 Ki = 458 nM T64765 CJW34M 11638322 Ki = 6.9 nM T64765 CR5QB1 11640354 Ki = 0.95 nM T64765 CMNV51 11640588 Ki = 0.16 nM T64765 CI2KZ1 11641036 Ki = 0.09688 nM T64765 CU25IV 11645244 Ki = 35 nM T64765 CSE96X 11645396 Ki = 0.1 nM T64765 C62YTU 11645731 Ki > 5000 nM T64765 C0M9NX 11646364 Ki = 0.37 nM T64765 CLR3P8 11646541 Ki = 1.25 nM T64765 CTZ1R2 11646905 Ki = 300 nM T64765 C24DVX 11647025 Ki = 0.2884 nM T64765 CA9QZ5 11647367 Ki = 8.3 nM T64765 C7XZ9J 11648391 Ki = 509 nM T64765 CFQD01 11652907 Ki = 140 nM T64765 CM5PG0 11653478 Ki = 0.85 nM T64765 CZV1D5 11653516 Ki = 4 nM T64765 CCGR62 11653567 Ki = 2 nM T64765 C8ZL6D 11653860 Ki = 9 nM T64765 C8I7UT 11654412 Ki = 516.7 nM T64765 CVH19Q 11654491 Ki = 125 nM T64765 CC59RQ 11655227 Ki = 13 nM T64765 CC36GP 11660512 Ki = 0.8 nM T64765 C4G9CM 11661358 IC50 = 3.2 nM T64765 CN7J5K 11661512 Ki = 11 nM T64765 CEYC43 11663122 Ki = 3 nM T64765 CT2AZ4 11663315 Ki = 25 nM T64765 CA76LI 11666530 Ki = 79 nM T64765 C6CMK7 11666852 Ki = 0.7 nM T64765 CPW3A8 11667985 Ki = 0.3125 nM T64765 C5WB3G 11668368 Ki = 2 nM T64765 CJSN27 11668594 Ki = 0.2812 nM T64765 C64GUF 11668827 Ki = 0.35 nM T64765 CG1Q3H 11668849 Ki = 3 nM T64765 CFEQ23 11669001 Ki = 0.56 nM T64765 CKT39R 11669791 Ki = 2 nM T64765 C1R6XC 11672850 Ki = 12.59 nM T64765 C1UGH0 11673377 Ki = 15.85 nM T64765 C7A0WS 11675333 Ki = 0.6875 nM T64765 CFQP90 11676381 Ki = 3.4 nM T64765 C3US8X 11676399 Ki = 0.29 nM T64765 CL3F6N 11679919 Ki = 7.943 nM T64765 CU5LI1 11679993 Ki = 3.162 nM T64765 CUSE05 11681731 Ki = 0.29 nM T64765 C8RA5V 11682068 Ki = 1.094 nM T64765 CPI01R 11682779 IC50 = 18 nM T64765 C6D0EL 11689049 Ki = 2.98 nM T64765 C1CB3H 11689509 EC50 = 1.585 nM T64765 C87TCD 11689687 Ki = 0.2812 nM T64765 CRXO13 11690171 Ki = 0.3 nM T64765 CL20PI 11690524 Ki = 8.7 nM T64765 CZ8TN6 11690910 Ki = 10 nM T64765 C3F9LC 11690966 Ki = 31 nM T64765 CU1LP9 11694543 Ki = 25.12 nM T64765 C21CHB 11694965 Ki = 0.5 nM T64765 C4EJ3V 11695488 Ki = 692 nM T64765 CEF73X 11695489 Ki = 0.11 nM T64765 CAKT97 11695753 Ki = 26 nM T64765 C6AIH4 11696359 IC50 = 43 nM T64765 CL8BO1 11696560 Ki = 0.31 nM T64765 CBG41V 11696718 Ki = 0.19 nM T64765 C3P0EV 11697383 IC50 = 43 nM T64765 CX7MT8 11697412 Ki = 21 nM T64765 C8K3OV 11698389 Ki = 0.74 nM T64765 C0SX3K 11701199 Ki = 100 nM T64765 CV4CL3 11702447 EC50 = 15.85 nM T64765 C5H4KG 11703337 IC50 = 33 nM T64765 CU5A6D 11703595 Ki = 0.74 nM T64765 C0UGV6 11703903 Ki = 34 nM T64765 C6G8WZ 11704156 IC50 = 10 nM T64765 C69MZL 11704938 Ki = 5.3 nM T64765 CA63UW 11708125 EC50 = 1.259 nM T64765 C78GTN 11709314 Ki = 10 nM T64765 C4UL2W 11709569 Ki = 0.08 nM T64765 C81JEA 11710150 Ki = 0.33 nM T64765 CXMH25 11710453 Ki = 0.1 nM T64765 C12EZH 11710694 Ki = 0.3 nM T64765 C9FBS2 11711947 Ki = 5.1 nM T64765 CJ0X7E 11716742 Ki = 200 nM T64765 CG0CD6 11717680 EC50 < 1 nM T64765 CI1C4Z 11718272 Ki = 6.8 nM T64765 CIH38K 11723422 Ki = 0.19 nM T64765 CD2ZL9 11724369 Ki = 15.85 nM T64765 CX5EM7 11725577 Ki = 129 nM T64765 CN32XC 11726879 Ki = 82 nM T64765 CLYO34 11728450 Ki = 530 nM T64765 C6E2PS 11739140 Ki = 1.5 nM T64765 CM6KJ7 11739735 Ki = 50.12 nM T64765 CIEN46 11741247 Ki = 0.1 nM T64765 CBLI40 11743550 Ki = 3 nM T64765 CRA6N7 11748896 Ki = 0.05 nM T64765 CEOK90 11759871 Ki = 66 nM T64765 C06EVL 11772496 Ki = 2.9 nM T64765 C7U5YP 11772738 Ki = 2.6 nM T64765 C62YRQ 11775426 Ki = 0.22 nM T64765 CI37HB 11776396 Ki = 21 nM T64765 CITX31 11776588 Ki = 87 nM T64765 C9LI8F 11779175 Ki = 86 nM T64765 CRX47N 11782172 Ki = 188 nM T64765 C7ODJ9 11788475 EC50 = 3.162 nM T64765 CH06GX 11794363 Ki = 30 nM T64765 CMDT64 11804748 EC50 > 0.0001 nM T64765 CP0TA5 11808122 Ki = 227 nM T64765 CGIC60 11808427 Ki = 50.12 nM T64765 CYC23D 11819221 EC50 = 1.318 nM T64765 C4XK5U 11822558 Ki = 334 nM T64765 CTA6K1 11824896 Ki = 7.8 nM T64765 CRD3P2 11825192 Ki = 890 nM T64765 CCAH67 11826604 Ki = 1.259 nM T64765 C4JIZ5 11829635 EC50 = 1410 nM T64765 C4Z3RD 11833907 Ki = 91 nM T64765 C0X7FJ 11846300 Ki = 9120.11 nM T64765 CXLW54 11948707 Ki > 10000 nM T64765 C32AQN 11949667 Ki = 0.1 nM T64765 CJ1YK2 11951972 EC50 = 7.943 nM T64765 C1CH2O 11957573 EC50 = 0.06918 nM T64765 CDH46N 11964510 Ki = 8.4 nM T64765 C38ACD 11973711 Ki = 0.17 nM T64765 CYEN98 11977494 Ki = 0.41 nM T64765 C03IKU 11977495 Ki = 1.64 nM T64765 CRDV32 11978735 Ki = 0.74 nM T64765 C7C8AJ 11978736 Ki = 0.82 nM T64765 CG96BD 11978737 Ki = 0.54 nM T64765 CN5W3V 11978858 Ki = 0.2 nM T64765 CW8T4V 11978859 Ki = 0.25 nM T64765 C1A2IB 12001199 Ki = 0.631 nM T64765 CBTO30 12214367 Ki = 345 nM T64765 C1Q9AY 12214369 Ki = 205 nM T64765 CURS31 12232304 Ki = 257.04 nM T64765 C4H1RC 12769844 EC50 = 1071.52 nM T64765 C2X3UC 13170764 IC50 = 2750 nM T64765 C1EO3M 13675122 Ki = 1.3 nM T64765 CAOF69 13995914 Ki = 543 nM T64765 C6PU9C 14097103 Ki = 2400 nM T64765 C7TH1U 14201494 Ki = 11000 nM T64765 CK8PA7 14201504 Ki = 80 nM T64765 C4CKI5 14201506 Ki = 1000 nM T64765 C3OFC7 14201508 Ki = 8000 nM T64765 CR4K2V 14201510 Ki = 4200 nM T64765 C8YSO7 14201512 Ki = 3300 nM T64765 CIZ8Q0 14201514 Ki = 1700 nM T64765 C7YMN9 14717864 Ki = 25.12 nM T64765 CF2GL7 14773975 Ki = 2000 nM T64765 C8BF2P 15254720 Ki = 398.11 nM T64765 C5S3CH 15288652 Ki > 1000 nM T64765 CW8R1S 15310636 Ki = 24 nM T64765 CHP9Y0 15604794 Ki = 4 nM T64765 CBE59I 15940927 Ki = 2.6 nM T64765 CA3YU5 15941764 Ki = 0.51 nM T64765 C18ZXI 15941903 Ki = 0.655 nM T64765 CMJ59Y 15941904 Ki = 0.057 nM T64765 C58TFK 15981911 Ki = 4 nM T64765 C6T5GH 15981916 Ki = 15 nM T64765 CJ7TI6 15981917 Ki = 13 nM T64765 CTU6F4 15982036 Ki = 13 nM T64765 CFPV59 15982037 Ki = 13 nM T64765 CIX70J 15982171 Ki = 13 nM T64765 CRN92T 15983453 Ki = 5 nM T64765 CYO4G3 15983454 Ki = 2 nM T64765 CMD02L 15983456 Ki = 1 nM T64765 C4SJF0 15983457 Ki = 4 nM T64765 CP94BW 15983458 Ki = 4 nM T64765 CM12TW 15983459 Ki = 12 nM T64765 C7X0TJ 15983575 Ki = 43 nM T64765 CP96DT 15983576 Ki = 90 nM T64765 CWQ59P 15983578 Ki = 8 nM T64765 CLV05C 15983579 Ki = 5 nM T64765 CF1H7C 15983580 Ki = 18 nM T64765 CY5U3T 15983703 Ki = 9 nM T64765 CEG95K 15983705 Ki = 23 nM T64765 CX2L9Q 15983706 Ki = 7 nM T64765 CDJ9B2 15983708 Ki = 2 nM T64765 C08HXO 15983836 Ki = 1 nM T64765 C8P2AR 15983838 Ki = 7 nM T64765 CE9Z5F 15983840 Ki = 13 nM T64765 C9K2MU 15983841 Ki = 7 nM T64765 CJ83YW 15984057 Ki = 0.3 nM T64765 CPR25X 15986917 Ki = 1.585 nM T64765 CRBP36 15987008 Ki = 0.7943 nM T64765 C5KW3L 15987108 Ki = 1 nM T64765 CF6S2D 15987282 Ki = 2.512 nM T64765 CXU15Z 15987451 Ki = 1.995 nM T64765 C6V3WY 15987452 Ki = 3.981 nM T64765 C0HKS9 16004748 Ki = 2 nM T64765 CA91OD 16005497 Ki = 5.7 nM T64765 C8V1IK 16005500 Ki = 4 nM T64765 CO0E2Y 16006089 Ki = 0.7 nM T64765 CDB1W5 16006612 Ki = 0.7 nM T64765 CQV08D 16006719 Ki = 1 nM T64765 C05CPW 16006947 Ki = 35 nM T64765 CU27FI 16049886 Ki = 17 nM T64765 CZC7L2 16049887 Ki = 14 nM T64765 CS8NZ0 16059780 Ki = 0.4467 nM T64765 C6V4HS 16059786 Ki = 4 nM T64765 CT6AL1 16061961 Ki = 323.59 nM T64765 C3ZKG6 16078981 EC50 = 48.98 nM T64765 CN6V3I 16082820 Ki > 1000 nM T64765 C52PUB 16082822 Ki = 34.4 nM T64765 C5ULI8 16082824 Ki = 203 nM T64765 C9Y8TA 16082826 Ki = 289 nM T64765 CV36OS 16082828 Ki = 8.4 nM T64765 CHTO30 16082831 Ki = 3.6 nM T64765 CJ1DV9 16082833 Ki = 5.3 nM T64765 CFJ53S 16082852 Ki = 88 nM T64765 CU4KB7 16082854 Ki > 1000 nM T64765 CW9SA4 16082856 Ki = 43.7 nM T64765 CRP4X3 16082858 Ki = 20.5 nM T64765 CT2NF0 16082860 Ki = 13.9 nM T64765 CIP39S 16082862 Ki > 1000 nM T64765 CT9B1U 16082864 Ki > 1000 nM T64765 C3YF6A 16082866 Ki > 1000 nM T64765 CFCK53 16112805 EC50 = 4 nM T64765 CJA65L 16119082 Ki = 1.047 nM T64765 C9BC4O 16119086 Ki = 1.698 nM T64765 C07RBX 16119587 Ki = 1.479 nM T64765 CFYL31 16122898 EC50 = 4 nM T64765 CS2HE1 16202149 Ki = 50.12 nM T64765 C1YWG6 16215415 Ki = 1040 nM T64765 C5EV2Z 16230818 IC50 > 10000 nM T64765 CZ2IS9 16660294 Ki > 10000 nM T64765 C0UZO6 16678214 EC50 = 25 nM T64765 C6K2ZB 16678514 Ki = 6 nM T64765 CTZE72 16678615 Ki = 14 nM T64765 CH0Q9T 16678616 Ki = 7 nM T64765 C80WKT 16678618 Ki = 6 nM T64765 CFEV50 16678619 Ki = 5 nM T64765 C4FUO7 16678620 Ki = 5 nM T64765 CDY08B 16678725 Ki = 46 nM T64765 C1N8IL 16679518 Ki = 25 nM T64765 CLI43T 16679519 Ki = 18 nM T64765 CA1JP4 16679520 Ki = 129 nM T64765 CDT2R3 16679611 Ki = 11 nM T64765 C0CF9G 16679612 Ki = 26 nM T64765 C8X6SN 16679614 Ki = 42 nM T64765 CH8A2G 16679616 Ki = 6 nM T64765 CBE9O8 16679617 Ki = 9 nM T64765 CQF5Y7 16679701 Ki = 17 nM T64765 CI9DM2 16679704 Ki = 21 nM T64765 CO03YT 16679705 Ki = 19 nM T64765 CGN61U 16679706 Ki = 34 nM T64765 CSK8N5 16679707 Ki = 31 nM T64765 C08XJA 16718567 IC50 = 5800 nM T64765 CDT5V8 16721129 Ki = 10 nM T64765 CQO3M8 16733807 Ki = 0.537 nM T64765 CYW3P2 16739387 Ki = 2 nM T64765 C4TFN0 16739412 EC50 = 2 nM T64765 CX6S1D 16739525 Ki = 1 nM T64765 CXBP47 16739577 EC50 = 6 nM T64765 CDK04H 16745305 Ki = 1160 nM T64765 CUG5B8 16747689 Ki = 0.6 nM T64765 CL4M3J 17931612 Ki = 236 nM T64765 CV8P5F 17962616 Ki = 12.88 nM T64765 CT0I8X 18428716 Ki = 9000 nM T64765 CG4CK9 18456143 Ki = 0.38 nM T64765 C73TRF 18456199 Ki = 1100 nM T64765 CA1Q3D 18456226 Ki = 89 nM T64765 CN46HY 18456227 Ki = 0.54 nM T64765 C81MQW 18456228 Ki = 0.86 nM T64765 CC63YZ 18456229 Ki = 480 nM T64765 CQWN78 18456232 Ki = 1.2 nM T64765 CCW85P 18456233 Ki = 34 nM T64765 CRE51J 18456234 Ki = 3.6 nM T64765 CG65WZ 18456235 Ki = 450 nM T64765 CX76WB 18456238 Ki = 1.2 nM T64765 C5WE8P 18456242 Ki = 8.3 nM T64765 CFG56D 18456243 Ki = 13.3 nM T64765 C40QGD 18456245 Ki = 4.4 nM T64765 CS29WF 18456246 Ki = 9.2 nM T64765 CD65ZG 18456437 Ki = 1.2 nM T64765 CV0EI2 18672441 Ki = 7.244 nM T64765 C1OE8D 18971393 IC50 = 7060 nM T64765 C9RK0S 20299674 Ki = 2.512 nM T64765 C7OLK5 20803169 Ki = 17 nM T64765 CB1N8D 20803171 Ki = 28 nM T64765 CX7RI6 20803174 Ki = 5400 nM T64765 C5JCZ6 21193534 Ki = 17 nM T64765 C3T5HF 21509921 Ki > 10000 nM T64765 C96TPD 21934845 Ki = 8.7 nM T64765 C6ACW2 22011795 Ki > 10000 nM T64765 CKM46E 22015607 Ki = 300 nM T64765 C7GVR9 22015611 Ki = 69 nM T64765 C0OKQ7 22015641 Ki = 10 nM T64765 CP7I6M 22015644 Ki = 15 nM T64765 C1B3GN 22016819 Ki = 812.83 nM T64765 C8ZTD3 22274462 Ki = 87 nM T64765 C51VOT 22274469 Ki = 12 nM T64765 CIU52R 22274472 Ki = 15.85 nM T64765 CWL61V 22274481 Ki = 3.9 nM T64765 CAF1L2 22274500 Ki = 8.8 nM T64765 CGCR83 22274513 Ki = 11.75 nM T64765 CD2CV9 22274699 Ki = 147.91 nM T64765 CFB23E 22390950 Ki = 0.5 nM T64765 C36WCQ 22493471 Ki = 0.871 nM T64765 C2USX1 22493482 Ki = 1.905 nM T64765 C8SGP4 22507782 Ki = 47 nM T64765 CH7D8A 23150257 Ki = 0.67 nM T64765 C3HD9T 23150285 Ki = 1.7 nM T64765 CYW7Q6 23150305 Ki = 10.4 nM T64765 C7ZUP3 23151143 IC50 = 103 nM T64765 C5MXI2 23151144 IC50 = 7 nM T64765 CCES43 23151160 IC50 = 1.2 nM T64765 CK7B0Q 23151166 IC50 > 1000 nM T64765 CX6DW5 23151169 IC50 = 1.2 nM T64765 C6QC2D 23151199 IC50 = 3.1 nM T64765 CGB8I7 23151202 IC50 = 5.8 nM T64765 CY8U0D 23151208 IC50 = 2 nM T64765 C3BP7D 23151209 IC50 = 0.55 nM T64765 CT78IA 23151210 IC50 = 0.84 nM T64765 C31KDO 23151223 IC50 = 8.6 nM T64765 CQ1K7H 23151224 Ki = 0.3125 nM T64765 CK4R0H 23151225 IC50 = 37 nM T64765 CU24MC 23151229 IC50 = 0.34 nM T64765 CM63GT 23151246 IC50 = 0.91 nM T64765 C47RDY 23151248 Ki = 0.7188 nM T64765 CU4DK0 23151250 IC50 = 1.5 nM T64765 C1D0AE 23151312 IC50 = 1.8 nM T64765 CE50PJ 23151323 IC50 = 1.8 nM T64765 C2KQ6N 23151327 IC50 = 1.3 nM T64765 CGJ78I 23151329 IC50 = 10 nM T64765 COPR89 23151331 Ki = 0.4688 nM T64765 C2NYB8 23151337 IC50 = 14 nM T64765 C12SUL 23151367 IC50 = 0.27 nM T64765 CR5OK1 23273673 Ki > 340 nM T64765 CL1YH7 23582308 Ki = 0.3162 nM T64765 C8VD3S 23624312 Ki = 1.8 nM T64765 C57MTL 23625757 Ki = 6 nM T64765 C0R8OI 23628252 EC50 = 0.2 nM T64765 C7MZX9 23649185 Ki = 1 nM T64765 C9PY4A 23725172 Ki = 1 nM T64765 CTM7A2 24729202 EC50 = 1513.56 nM T64765 C0B8DK 24738376 Ki = 33.11 nM T64765 C84RTS 24743472 Ki = 229 nM T64765 CVGT95 24743473 Ki = 54.95 nM T64765 C7TM6E 24743474 Ki = 3.236 nM T64765 CSA1P6 24743542 Ki = 4.898 nM T64765 CQ61DA 24743546 Ki = 5.888 nM T64765 CKU8E6 24743580 Ki = 1.51 nM T64765 C9RTG5 24743584 Ki = 10.7 nM T64765 C7H3FR 24743745 Ki = 26.3 nM T64765 CQ29UD 24743746 Ki = 25.1 nM T64765 CL82UB 24743987 Ki = 6.607 nM T64765 CHO9S8 24743988 Ki = 42.66 nM T64765 CHW15A 24743989 Ki = 70.79 nM T64765 CB10VA 24743990 Ki = 549.54 nM T64765 CRN13C 24748804 Ki = 0.7943 nM T64765 CTIF10 24748806 Ki = 3.162 nM T64765 CMJU59 24748889 Ki = 1.995 nM T64765 CB6R3K 24748890 Ki = 0.631 nM T64765 C5EQ8T 24748892 Ki = 3.981 nM T64765 CUMP36 24748894 Ki = 2.512 nM T64765 C1XN4V 24748896 Ki = 6.31 nM T64765 CFR1S3 24748988 Ki = 3.981 nM T64765 CG43ZS 24748989 Ki = 5.012 nM T64765 C96KDH 24748992 Ki = 0.631 nM T64765 CH8N1W 24748993 Ki = 0.5012 nM T64765 CQF29T 24749076 Ki = 3.162 nM T64765 CU0GX7 24749078 Ki = 5.012 nM T64765 CGD2I7 24749080 Ki = 3.162 nM T64765 CB8DF0 24749082 Ki = 2.512 nM T64765 C9XS6U 24749083 Ki = 3.981 nM T64765 CKVA89 24749182 Ki = 1.995 nM T64765 CRGJ52 24749183 Ki = 3.162 nM T64765 C13GRZ 24749184 Ki = 1 nM T64765 C8ZE6H 24749185 Ki = 0.631 nM T64765 CG9I8K 24749186 Ki = 1.259 nM T64765 CF8W2P 24749291 Ki = 1.585 nM T64765 CTB38H 24749292 Ki = 0.3162 nM T64765 CET71X 24749293 Ki = 2.512 nM T64765 CAE9S7 24749294 Ki = 0.7943 nM T64765 CKV83Y 24749295 Ki = 2.512 nM T64765 C6S0OJ 24749401 Ki = 3.981 nM T64765 CSG9V8 24749508 Ki = 1.585 nM T64765 CWTB59 24749606 Ki = 3.981 nM T64765 CLFS68 24749607 Ki = 1.995 nM T64765 CHYC87 24749609 Ki = 2.512 nM T64765 CY53AF 24749610 Ki = 7.943 nM T64765 CT93NP 24749721 Ki = 3.162 nM T64765 C7EGL2 24749724 Ki = 3.162 nM T64765 CW19JN 24749726 Ki = 7.943 nM T64765 CI6W7D 24749841 Ki = 0.631 nM T64765 CV20EP 24749844 Ki = 1.585 nM T64765 CYI79E 24749958 Ki = 0.7943 nM T64765 CGT53R 24749959 Ki = 3.981 nM T64765 C20QND 24749960 Ki = 0.631 nM T64765 CSXA65 24749962 Ki = 0.7943 nM T64765 CNOX23 24750086 Ki = 3.162 nM T64765 C1XRY9 24750087 Ki = 0.7943 nM T64765 C89WKU 24750088 Ki = 10 nM T64765 C6JRO5 24756897 EC50 = 3 nM T64765 C8GE2F 24770906 Ki = 4.7 nM T64765 C6Y1QZ 24770907 Ki = 5.5 nM T64765 C5PV4C 24770908 Ki = 4.3 nM T64765 CTM7F5 24770909 Ki = 17 nM T64765 C40JCH 24770911 Ki = 31 nM T64765 C97IRG 24770912 Ki = 40 nM T64765 CSG29Y 24770965 Ki = 9000 nM T64765 CRIF10 24770966 Ki = 860 nM T64765 C40QCZ 24771013 Ki = 29 nM T64765 CLAR45 24771015 Ki = 3.7 nM T64765 CP8CA9 24771016 Ki = 34 nM T64765 C7LQD8 24771017 Ki = 79 nM T64765 CKB2Q9 24771071 Ki = 2.3 nM T64765 C5RD6X 24771241 Ki = 78 nM T64765 C5OV6F 24771243 Ki = 230 nM T64765 CJ92VA 24771244 Ki = 100 nM T64765 C0JO5H 24771245 Ki = 260 nM T64765 C8Q2CL 24771304 Ki = 110 nM T64765 CV04EK 24771305 Ki = 73 nM T64765 CRCO59 24771307 Ki = 13 nM T64765 CXL49M 24771308 Ki = 12 nM T64765 CKOS32 24771362 Ki = 10 nM T64765 CV3P7F 24771363 Ki = 7.6 nM T64765 CU3M8O 24771364 Ki = 18 nM T64765 C4IPH3 24771367 Ki = 25 nM T64765 CH5DC3 24771416 Ki = 4.4 nM T64765 CFDM36 24771417 Ki = 430 nM T64765 C4WUI2 24771418 Ki = 17 nM T64765 C56EJY 24771419 Ki = 1 nM T64765 C6H9WM 24771420 Ki = 59 nM T64765 CY49MU 24771522 Ki = 16 nM T64765 COGS63 24771524 Ki = 4.1 nM T64765 C06DCW 24771574 Ki = 1040 nM T64765 C3U7NP 24771575 Ki = 160 nM T64765 CYPK78 24771576 Ki = 430 nM T64765 CJ31PE 24771627 Ki = 1.5 nM T64765 CUW8I3 24771629 Ki = 10 nM T64765 C5I9SQ 24771740 Ki = 5.5 nM T64765 CJ9W6U 24771741 Ki = 2.9 nM T64765 CKCQ70 24783527 Ki = 2.1 nM T64765 C5Z1AB 24798144 Ki = 24 nM T64765 CUX7C3 24803316 Ki = 0.3981 nM T64765 C1QTN4 24803480 Ki = 7.943 nM T64765 CTU67D 24803482 Ki = 0.2512 nM T64765 C31QHW 24803483 Ki = 0.3981 nM T64765 C3RYC2 24803638 Ki = 0.3162 nM T64765 CI4EA6 24803639 Ki = 0.3981 nM T64765 CJ07ES 24803641 Ki = 0.5012 nM T64765 C04KHJ 24803797 Ki = 3.981 nM T64765 CY26TH 24803798 Ki = 0.2512 nM T64765 C50BOH 24803799 Ki = 1.995 nM T64765 C2AKX9 24804150 Ki = 0.5623 nM T64765 CSZG69 24825510 Ki = 3.981 nM T64765 C7TPA1 24825511 Ki = 154.88 nM T64765 C61ZJM 24825512 Ki = 40.74 nM T64765 CU9C5R 24825513 Ki = 426.58 nM T64765 CLB5M8 24825514 Ki = 32.36 nM T64765 C8DQR0 24825515 Ki = 4.467 nM T64765 CYFC27 24825517 Ki = 1737.8 nM T64765 C41FJM 24825519 Ki = 2511.89 nM T64765 CSYK46 24825520 Ki = 416.87 nM T64765 C0KG2Y 24825521 Ki = 537.03 nM T64765 CIM1V9 24825522 Ki = 1.259 nM T64765 C8S7TO 24825523 Ki = 39.81 nM T64765 CGNO06 24825524 Ki = 56.23 nM T64765 CXO2M4 24825525 Ki = 707.95 nM T64765 CCWS85 24825526 EC50 = 79.43 nM T64765 C0DHK4 24825527 Ki = 2511.89 nM T64765 C2BNX5 24825718 Ki = 2.5 nM T64765 CDC91N 24839550 Ki < 10000 nM T64765 CY21RE 24841480 Ki = 6000 nM T64765 C50XIV 24855884 Ki = 1.8 nM T64765 CJTY89 24855886 Ki = 2 nM T64765 C79FCO 24855918 Ki = 1 nM T64765 CJAC42 24855949 Ki = 0.8 nM T64765 C1SVD5 24855952 Ki = 4.1 nM T64765 CYQS46 24855953 Ki = 1.4 nM T64765 CGC54I 24855977 Ki = 1.2 nM T64765 CAF5W4 24855979 Ki = 1.5 nM T64765 C96KWD 24855980 Ki = 1.4 nM T64765 CEV3S9 24855981 Ki = 1.1 nM T64765 C3A6SC 24856010 Ki = 0.7 nM T64765 C5T6WF 24856012 Ki = 0.8 nM T64765 C2BG9R 24856014 Ki = 1 nM T64765 CS1VR8 24856015 Ki = 5.5 nM T64765 CG07AV 24856046 Ki = 2.1 nM T64765 C67OXE 24856047 Ki = 1 nM T64765 CW0J7T 24856048 Ki = 2 nM T64765 CE2UI4 24856107 Ki = 1.1 nM T64765 C48LYD 24856108 Ki = 1 nM T64765 CU34QD 24884554 Ki = 1 nM T64765 CNF2E4 24885663 Ki = 4.266 nM T64765 CJO97K 24885890 Ki = 3.162 nM T64765 C0FUC5 24886365 Ki = 1 nM T64765 C9A2NF 24890939 Ki = 23 nM T64765 CM7F6V 24896761 Ki = 0.4 nM T64765 C7J4ZQ 24900259 IC50 = 0.7 nM T64765 CZPW63 24936097 Ki = 14 nM T64765 CQ52SD 24936098 Ki = 0.39 nM T64765 C1GAD9 24946664 Ki = 7.7 nM T64765 CF26PB 24946667 Ki = 2.4 nM T64765 C9W1EB 24946668 Ki = 3.4 nM T64765 CWK21C 24947199 Ki = 2.7 nM T64765 CDI10X 24947200 Ki = 3.3 nM T64765 CO2TD9 24947376 Ki = 0.9 nM T64765 CIG62P 24947377 Ki = 0.2 nM T64765 CI6TP1 24947378 Ki = 0.7 nM T64765 CSL93K 24947379 Ki = 1 nM T64765 CY9X8Z 24947380 Ki = 1.7 nM T64765 C20BSY 24947381 Ki = 0.9 nM T64765 C3H5PJ 24947569 Ki = 29 nM T64765 CUM1C3 24947570 Ki = 1 nM T64765 CERD40 24947571 Ki = 1.7 nM T64765 CB2U7X 24947572 Ki = 0.9 nM T64765 CQ7Z6F 24947573 Ki = 0.7 nM T64765 CEGC24 24947574 Ki = 0.9 nM T64765 CSJ5I4 24947575 Ki = 1 nM T64765 C4Y7FP 24947750 Ki = 2.2 nM T64765 CA8VN2 24947751 Ki = 4.3 nM T64765 CYGT57 24947752 Ki = 1.1 nM T64765 CL60YE 24947753 Ki = 1.1 nM T64765 C1FSB7 24947760 Ki = 5 nM T64765 CFJ4O7 24947761 Ki = 1.3 nM T64765 CEW8C3 24947936 Ki = 14 nM T64765 CVZ7K9 24947937 Ki = 6.8 nM T64765 C72EWS 24947938 Ki = 15 nM T64765 C8TKG2 24947939 Ki = 37 nM T64765 C6BIR1 24947941 Ki = 21 nM T64765 C06TLI 24948121 Ki = 11 nM T64765 C2OK6I 24948317 Ki = 0.8 nM T64765 C9WPU6 24948318 Ki = 0.7 nM T64765 C0BL9R 24948319 Ki = 0.8 nM T64765 C8MU7D 24948320 Ki = 2.3 nM T64765 CJ0M6T 24948507 Ki = 1 nM T64765 CYL4U5 24948945 Ki = 0.25 nM T64765 CQU27P 24948946 Ki = 0.2188 nM T64765 CRJ08Z 24948948 Ki = 0.625 nM T64765 CC17EO 24950873 Ki = 1.156 nM T64765 C6Z9PO 24951035 IC50 = 2.2 nM T64765 CV0PG1 24951036 IC50 = 4.3 nM T64765 CWQ7Z3 24951037 IC50 = 20 nM T64765 CB03UR 24951038 IC50 = 0.72 nM T64765 CH36LE 24951189 IC50 = 41 nM T64765 C02ADX 24951191 Ki = 0.3125 nM T64765 C7WE9M 24951192 Ki = 0.625 nM T64765 CVT49O 24951193 Ki = 0.4062 nM T64765 C7DGE0 24951348 Ki = 0.5 nM T64765 C9GA3W 24951349 Ki = 0.3125 nM T64765 COW04Z 24951350 Ki = 0.6875 nM T64765 CHD86F 24951351 Ki = 0.2188 nM T64765 C2XUP4 24963805 Ki = 11 nM T64765 C6DW3J 24964157 Ki = 1.7 nM T64765 CQ42YZ 24964158 Ki = 11 nM T64765 C4P5AD 24964159 Ki = 11 nM T64765 CP6SX7 24964160 Ki = 7 nM T64765 CP53AB 24964161 Ki = 5.7 nM T64765 C3YXJ9 24964162 Ki = 7.3 nM T64765 CZV16S 24964163 Ki = 3 nM T64765 C2PA7D 24964521 Ki = 31 nM T64765 CFPU09 24964522 Ki = 3 nM T64765 CYK2Q6 24964523 Ki = 52 nM T64765 CNU2L1 24964524 Ki = 17 nM T64765 C2L0PV 24964525 Ki = 17 nM T64765 C1X3LT 24964877 Ki = 9.7 nM T64765 CN7B3D 24964878 Ki = 864 nM T64765 C8KID6 24964879 Ki = 93 nM T64765 CA3T8S 24965234 Ki = 1867 nM T64765 COH49Y 24965236 Ki = 13 nM T64765 CK2I8F 24965237 Ki = 6 nM T64765 C9PVS1 24965238 Ki = 14 nM T64765 CY0IN2 24965589 Ki = 4.7 nM T64765 CL56YC 24965590 Ki = 5.2 nM T64765 C1SUL8 24965930 Ki = 423 nM T64765 CWA0R4 24978528 Ki = 7.943 nM T64765 C4PU9I 24992189 Ki = 14 nM T64765 CGRO26 24992190 Ki = 3.4 nM T64765 CWAC54 24992193 Ki = 1.9 nM T64765 CKMB97 24992194 Ki = 3 nM T64765 CP14IG 24992516 Ki = 8.7 nM T64765 CL83OS 24992519 Ki = 1.4 nM T64765 CK7X4Q 24992520 Ki = 26 nM T64765 C16SVM 24992849 Ki = 6.3 nM T64765 CVX0T7 24992850 Ki = 15 nM T64765 CRO45L 24992851 Ki = 5.9 nM T64765 CTH32Z 24992852 Ki = 1.8 nM T64765 CO9F7A 24992853 Ki = 6.5 nM T64765 CKI14H 24992854 Ki = 35 nM T64765 CS3CD7 24993174 Ki = 12 nM T64765 C62OQY 24993175 Ki = 34 nM T64765 CZA68B 24993176 Ki = 3.7 nM T64765 C8KIP6 24993178 EC50 = 0.8 nM T64765 CWM6J4 24993179 Ki = 7.1 nM T64765 C58WOG 24993499 Ki = 5.1 nM T64765 CD8U2B 24993500 EC50 = 1.1 nM T64765 C60TYB 24993502 Ki = 9.8 nM T64765 CCDF20 24994127 EC50 = 0.7 nM T64765 CKXQ41 24994432 Ki = 12 nM T64765 CV7N9Y 24994433 Ki = 7.1 nM T64765 CW8J0F 24994438 Ki = 83 nM T64765 CA82IM 24994744 Ki = 3.1 nM T64765 COR42A 24994745 Ki = 6.2 nM T64765 CR50CS 24995678 Ki = 15 nM T64765 C51SKE 24995679 Ki = 2.7 nM T64765 CPLJ75 24995680 Ki = 11 nM T64765 C4QN1A 24995681 Ki = 4.4 nM T64765 CJM8R0 24996322 Ki = 1.7 nM T64765 CK5LM1 24996644 EC50 = 1.1 nM T64765 CFDQ56 24996645 Ki = 3 nM T64765 CTL2D0 24996647 Ki = 2 nM T64765 C63FIB 24996648 Ki = 3 nM T64765 C0L8SV 24996965 Ki = 15 nM T64765 CE72ZO 24996966 Ki = 12 nM T64765 CUN71B 24996967 Ki = 9.9 nM T64765 CLSJ69 25030982 Ki = 390 nM T64765 CB1VG2 25030983 Ki = 17 nM T64765 CBV91O 25031068 Ki = 10 nM T64765 C6Q2AM 25031073 Ki = 5 nM T64765 CSI78Z 25032211 Ki = 440 nM T64765 C4MKP1 25032212 Ki = 3 nM T64765 C84NVG 25032264 Ki = 100 nM T64765 CT1IH5 25032267 Ki = 65 nM T64765 CN5PV0 25053284 Ki = 60.26 nM T64765 C2E9AS 25053285 Ki = 39.8 nM T64765 C5XPK9 25053286 Ki = 3.31 nM T64765 C1OPU7 25053347 Ki = 1.66 nM T64765 C45GSV 25053348 Ki = 50.1 nM T64765 CPY37G 25053349 Ki = 23.4 nM T64765 CXYF30 25053350 Ki = 19 nM T64765 C2G1JK 25053351 Ki = 0.2089 nM T64765 C01PUM 25053421 Ki = 1.148 nM T64765 C0H8DL 25053422 Ki = 19.7 nM T64765 CKVX12 25053423 Ki = 109.65 nM T64765 CNIE12 25053424 Ki = 12.3 nM T64765 CMZU43 25053425 Ki = 16.2 nM T64765 C5GJO7 25053485 Ki = 60.26 nM T64765 CE42WS 25053486 Ki = 30.9 nM T64765 C2K6WT 25053487 Ki = 7.76 nM T64765 C08VHD 25053488 Ki = 0.37 nM T64765 CV8W3D 25053489 Ki = 1.62 nM T64765 C8VOT9 25059091 Ki = 43 nM T64765 C8YK1V 25061409 Ki = 2 nM T64765 C54YBL 25061410 Ki = 1.4 nM T64765 CAGR71 25061412 Ki = 15 nM T64765 CL1UM3 25061663 Ki = 4.9 nM T64765 C90INA 25061920 Ki = 12 nM T64765 CM3FW6 25061923 Ki = 1.6 nM T64765 CXG08V 25061924 Ki = 2.8 nM T64765 CC14AS 25061926 Ki = 27 nM T64765 C8SJ9L 25062200 Ki = 1.9 nM T64765 C30DIE 25062467 Ki = 88 nM T64765 CEA69Y 25062471 Ki = 180 nM T64765 C3NQ5I 25062473 Ki = 4900 nM T64765 CGF15E 25062737 Ki = 88 nM T64765 CWIF74 25062740 Ki = 240 nM T64765 CM83VQ 25067563 Ki = 4.7 nM T64765 CC6NZ8 25095678 Ki = 1.3 nM T64765 C51OJR 25099115 IC50 = 0.54 nM T64765 CMX36H 25107505 Ki > 10000 nM T64765 C7NJ1B 25109291 Ki = 933.25 nM T64765 C0QOD8 25117760 IC50 = 12 nM T64765 CYP71T 25118123 IC50 = 1100 nM T64765 CH57JF 25118124 Ki = 11 nM T64765 C6C0HA 25118125 Ki = 3 nM T64765 CM2G5L 25118126 Ki = 65 nM T64765 C4DMZ5 25118127 Ki = 1.4 nM T64765 CUVK38 25118474 Ki = 8.4 nM T64765 CU9C3A 25118476 IC50 = 16 nM T64765 CXE6T1 25118477 IC50 = 10 nM T64765 C9Z4KB 25118479 IC50 = 19 nM T64765 C8NVJ5 25118830 IC50 = 66 nM T64765 CNIT95 25118831 Ki = 103 nM T64765 CY18PX 25119191 Ki = 55 nM T64765 CDO7F3 25120248 Ki = 17 nM T64765 C4AX6K 25120607 Ki = 252 nM T64765 CS6O1Q 25120608 Ki = 6.7 nM T64765 CNZ6R7 25120609 Ki = 32 nM T64765 CE3HK2 25120611 Ki = 26 nM T64765 C2G0BK 25120953 Ki = 1.6 nM T64765 CLV98T 25120954 Ki = 2.7 nM T64765 C28XUO 25120956 Ki = 7.3 nM T64765 CR2D3W 25122009 Ki = 1.8 nM T64765 CN65EI 25122012 Ki = 144 nM T64765 CI6WZ1 25122747 Ki = 197 nM T64765 CCB62X 25122748 Ki = 19 nM T64765 CDMT45 25122749 Ki = 26 nM T64765 C30YQW 25126154 Ki = 1.5 nM T64765 CML6G5 25128822 Ki = 9772.37 nM T64765 C7QMJ4 25129169 Ki = 2238.72 nM T64765 C7JU1L 25130576 Ki = 933.25 nM T64765 C4S5QV 25139031 IC50 = 740 nM T64765 C5FS6U 25139032 IC50 = 60 nM T64765 C9DQ8L 25139490 IC50 = 3 nM T64765 CWL9E2 25139491 IC50 = 4.2 nM T64765 C3XJM1 25139625 IC50 = 10 nM T64765 CKLC61 25139757 IC50 = 1.5 nM T64765 C4N1YF 25139758 IC50 = 1.7 nM T64765 C4R6JL 25141139 Ki = 100 nM T64765 C5ME9J 25147728 Ki = 1.995 nM T64765 C8D7HZ 25149335 EC50 = 2.45 nM T64765 C4GC8J 25149708 EC50 = 1.64 nM T64765 C6NAC0 25149712 EC50 = 2.512 nM T64765 CJVM09 25156194 Ki = 0.15 nM T64765 C0TI3Z 25156476 Ki = 3.2 nM T64765 CMX1W0 25156477 Ki = 1.8 nM T64765 C24UVQ 25156478 Ki = 0.25 nM T64765 C8AYP4 25156480 Ki = 1 nM T64765 C1HG2K 25156481 Ki = 5.1 nM T64765 CKP4R2 25156482 Ki = 230 nM T64765 CBM05I 25156750 Ki = 0.93 nM T64765 C3QT7F 25156751 Ki = 0.89 nM T64765 CJPO67 25156752 Ki = 0.98 nM T64765 CAQE42 25211254 Ki = 1.9 nM T64765 C78HME 25212275 Ki = 0.042 nM T64765 CE6Z9I 25212276 Ki = 0.358 nM T64765 CJ1Z9H 25216680 Ki = 1 nM T64765 C6EO8B 25216683 Ki = 1 nM T64765 CYAL71 25217063 Ki = 6 nM T64765 CJW54O 25217064 Ki = 0.8 nM T64765 CV1YR5 25217066 Ki = 18 nM T64765 CAO6R0 25217067 Ki = 5.7 nM T64765 CXK8C2 25217299 Ki = 3.1 nM T64765 CA8RO1 25217406 Ki = 3.2 nM T64765 CLHN01 25217407 Ki = 1.3 nM T64765 CT67WG 25217408 Ki = 1.6 nM T64765 C9D8TU 25217517 Ki = 11 nM T64765 CL2N5G 25217518 Ki = 9 nM T64765 CB3F9J 25217519 Ki = 8.1 nM T64765 C05NCT 25217636 Ki = 14.1 nM T64765 C8NZL4 25217637 Ki = 28.4 nM T64765 CQE8D6 25217638 Ki = 14.9 nM T64765 C0ANW9 25217639 Ki = 3.4 nM T64765 C16WTA 25217640 Ki = 11.4 nM T64765 C9BGS6 25217760 Ki = 11.6 nM T64765 C2WN4U 25217761 Ki = 3.9 nM T64765 C5WI0J 25217762 Ki = 6.4 nM T64765 CB21JO 25217764 Ki = 9.3 nM T64765 CG0BR7 25217887 Ki = 7.7 nM T64765 CXWM05 25217888 Ki = 2.4 nM T64765 C5N7UR 25217890 Ki = 21.7 nM T64765 C4RI6Q 25217891 Ki = 6.9 nM T64765 C9UGR4 25217893 Ki = 7.8 nM T64765 CJ0Y7P 25218014 Ki = 12.7 nM T64765 CW7RJ2 25218015 Ki = 1.2 nM T64765 CSX86U 25218016 Ki = 2.1 nM T64765 CT3LJ6 25218017 Ki = 0.8 nM T64765 C08NBX 25218019 Ki = 1.2 nM T64765 C1XQ6U 25218020 Ki = 0.6 nM T64765 CJIU87 25218140 Ki = 0.3 nM T64765 C0VI2J 25218142 Ki = 2.4 nM T64765 C1T3LR 25218143 Ki = 1.9 nM T64765 C8RCG2 25218267 Ki = 2.7 nM T64765 C6VNQ4 25218268 Ki = 1.2 nM T64765 C0ONJ9 25218269 Ki = 1.3 nM T64765 CU63JR 25218271 Ki = 1.9 nM T64765 CPI03N 25218397 Ki = 0.9 nM T64765 C4GSU5 25218398 Ki = 2.1 nM T64765 CL1R3Q 25218401 Ki = 0.2 nM T64765 C5CFH0 25218402 Ki = 6 nM T64765 CV29RL 25229699 IC50 = 0.1 nM T64765 C6VSX9 25263864 IC50 = 1.2 nM T64765 C03SUJ 25263865 IC50 = 0.9 nM T64765 CNCD39 25263866 IC50 = 3.1 nM T64765 C16ARL 25263867 IC50 = 1.1 nM T64765 CZ9E8H 25263989 IC50 = 0.1 nM T64765 C6IA9Q 25263990 IC50 = 0.2 nM T64765 CTFN54 25263991 IC50 = 0.2 nM T64765 CCFD64 25263992 IC50 = 0.2 nM T64765 C1YV5R 25264117 IC50 = 1.1 nM T64765 CQ5V9F 25264118 IC50 = 1.1 nM T64765 CR64VD 25264119 IC50 = 0.3 nM T64765 CFV1P6 25264121 IC50 = 0.2 nM T64765 C5QZY6 25264122 IC50 = 0.8 nM T64765 C8NHL5 25264260 IC50 = 1.1 nM T64765 CV4U6C 25264261 IC50 = 0.4 nM T64765 C9GCH0 25264262 IC50 = 0.5 nM T64765 CES94Q 25264263 IC50 = 2.3 nM T64765 C5E3ZH 25265089 Ki = 0.1 nM T64765 C5BNH3 25265516 EC50 = 0.9 nM T64765 C47WLU 27160619 Ki = 22.7 nM T64765 CR6Q3D 34598448 IC50 = 10000 nM T64765 CJ8V4H 34681379 IC50 > 10000000 nM T64765 CA4WZ7 35275893 IC50 = 40.5 nM T64765 C2TKY0 35476763 IC50 > 10000 nM T64765 CW04EV 40011786 Ki = 100 nM T64765 CIC89O 42604517 Ki = 3.2 nM T64765 C5SJB9 42623567 EC50 = 25.12 nM T64765 C7SQE1 42623731 EC50 = 12.59 nM T64765 CN7KY1 42624149 Ki = 670 nM T64765 CIJ52Y 42625222 EC50 = 15.85 nM T64765 CR7LN9 42625223 EC50 = 10.96 nM T64765 C8G7QX 42625303 EC50 = 1.585 nM T64765 C75WJN 42625304 EC50 = 1.413 nM T64765 C0BW6J 42625384 EC50 = 3.631 nM T64765 CID4J1 42625386 EC50 = 1.585 nM T64765 CRO42D 42629969 Ki = 27.9 nM T64765 CE7RV9 42630823 Ki < 25 nM T64765 CEZU81 44072806 Ki = 6118 nM T64765 C9HPN4 44158482 IC50 = 12 nM T64765 CQH86Y 44158485 IC50 = 58.5 nM T64765 C9AZM8 44158486 IC50 = 32 nM T64765 CZG07X 44158590 IC50 = 28 nM T64765 C3RKI7 44158698 IC50 = 0.4 nM T64765 C90CDL 44158699 IC50 = 0.9 nM T64765 C16AUE 44158811 IC50 = 0.2 nM T64765 CVN2U8 44158813 IC50 = 47 nM T64765 CO60AP 44159044 IC50 = 41 nM T64765 C7EJK3 44159045 IC50 = 6.5 nM T64765 C9X7BQ 44159046 IC50 = 51 nM T64765 CBG95A 44159047 IC50 = 0.4 nM T64765 CV6M8R 44159170 IC50 = 17 nM T64765 CVQ89M 44159172 IC50 = 42 nM T64765 C7AO3V 44159173 IC50 = 119 nM T64765 C6NA7M 44159287 IC50 = 102 nM T64765 CSL9R4 44159519 IC50 = 551 nM T64765 C7JRG6 44159523 IC50 = 0.6 nM T64765 C52EQI 44159636 IC50 = 0.5 nM T64765 C4O6KW 44159637 IC50 = 6.8 nM T64765 C9RC2Z 44159640 IC50 = 4.6 nM T64765 C1C2DH 44159759 IC50 = 1.6 nM T64765 CKOP76 44159760 IC50 = 115 nM T64765 CZ5NK7 44159763 IC50 = 33 nM T64765 CZ4P8Q 44159883 IC50 = 21 nM T64765 CY9F6U 44159887 IC50 = 98 nM T64765 CN6OI8 44160009 IC50 = 58 nM T64765 CAC2U0 44160010 IC50 = 1.2 nM T64765 CZA9M8 44160131 IC50 = 0.7 nM T64765 C5GYS4 44160248 IC50 = 1.6 nM T64765 C3G0JL 44184899 EC50 < 1 nM T64765 CSXG15 44184902 Ki = 1 nM T64765 CW9BU5 44184903 EC50 = 9 nM T64765 C5AC0D 44184949 EC50 = 2 nM T64765 C3WP4U 44185183 Ki = 86 nM T64765 CQJF53 44185243 EC50 = 112 nM T64765 C14BUY 44185245 Ki = 4 nM T64765 CYL93A 44187557 Ki = 6.31 nM T64765 C6P7EH 44211094 EC50 = 794.33 nM T64765 CK2GH7 44215409 Ki = 308 nM T64765 CP52BC 44215411 Ki = 40 nM T64765 CJS6F8 44215412 Ki = 11 nM T64765 CKLU60 44221502 Ki = 323.59 nM T64765 CF20NJ 44221503 Ki = 100 nM T64765 CG50TW 44221505 Ki < 1000 nM T64765 CM3QE5 44221508 Ki = 114.82 nM T64765 C26RAZ 44221712 Ki < 1000 nM T64765 CBVW68 44221713 Ki = 15.49 nM T64765 C6W9VE 44221714 Ki = 14.45 nM T64765 CH4G9N 44221717 Ki = 549.54 nM T64765 CBDU07 44221718 Ki = 13.18 nM T64765 CO4MD8 44221719 Ki = 512 nM T64765 C3OXF4 44221914 Ki = 12.3 nM T64765 CFYE69 44221915 Ki = 181.97 nM T64765 CW9SX8 44221916 Ki = 4.14 nM T64765 CRK71W 44221917 Ki = 20.4 nM T64765 C64WXB 44224176 Ki = 30 nM T64765 CL2IE8 44231618 Ki = 63.1 nM T64765 C3OA5J 44231733 Ki = 295.12 nM T64765 CP5MX1 44231735 Ki = 104.71 nM T64765 C0Z3PB 44243713 Ki = 14.45 nM T64765 CDOA12 44249906 EC50 = 17 nM T64765 C8P2LE 44250288 Ki = 0.4 nM T64765 CMD87L 44254048 Ki = 2.512 nM T64765 CXA10D 44254307 Ki = 5.012 nM T64765 CQBA78 44269558 Ki = 33 nM T64765 CZV6S4 44269697 Ki = 70 nM T64765 C5YIJ9 44269722 Ki = 3.6 nM T64765 C28URK 44275408 Ki = 18.2 nM T64765 CJ9G0A 44275409 Ki = 3.467 nM T64765 C9PHU6 44275419 Ki = 6.918 nM T64765 CJ5G8C 44275443 Ki = 0.6026 nM T64765 CZ6JS0 44275454 Ki = 5.129 nM T64765 CMZ78L 44275455 Ki = 229.09 nM T64765 CEL7B6 44275464 Ki = 1.122 nM T64765 CQ4X7K 44275478 Ki = 24.55 nM T64765 C1A5RO 44275495 Ki = 2.138 nM T64765 CWD95Y 44275496 Ki = 9.772 nM T64765 CK1I0D 44275508 Ki = 0.7762 nM T64765 CXZ96U 44275528 Ki = 6.166 nM T64765 C4LPN0 44275530 Ki = 37.15 nM T64765 CCZP76 44275533 Ki = 3.715 nM T64765 CYW7F1 44275534 Ki = 8.318 nM T64765 CF2NS6 44275538 Ki = 4.677 nM T64765 CT2LF1 44275542 Ki = 2.089 nM T64765 C0DTA1 44275543 Ki = 8.128 nM T64765 C61YFK 44275553 Ki = 0.9772 nM T64765 CY70TP 44275558 Ki = 6.457 nM T64765 CT51VC 44275562 Ki = 11.22 nM T64765 CICE54 44275563 Ki = 4.365 nM T64765 C0DW2J 44275597 Ki = 16.22 nM T64765 CS7EI6 44275619 Ki = 0.7762 nM T64765 CK60XA 44275620 Ki = 4.786 nM T64765 C41HJB 44275637 Ki = 8.128 nM T64765 C4HGI1 44275638 Ki = 6.918 nM T64765 C7DXL0 44275646 Ki = 32.36 nM T64765 CX8OY3 44275668 Ki = 7.244 nM T64765 C2ZA8O 44275749 Ki = 38.9 nM T64765 CUHT09 44275760 Ki = 109.65 nM T64765 C6K8ZH 44275761 Ki = 0.8511 nM T64765 C5YGL0 44275774 Ki = 40.74 nM T64765 CDE37G 44275781 Ki = 2.399 nM T64765 C3ZDJ1 44275793 Ki = 0.6918 nM T64765 CNZ4T8 44275797 Ki = 3.631 nM T64765 CQH7B4 44275798 Ki = 6.457 nM T64765 CE20CZ 44275807 Ki = 0.4898 nM T64765 C3IC9G 44275828 Ki = 3.02 nM T64765 CAH01T 44275830 Ki = 23.44 nM T64765 CC9D2J 44275843 Ki = 10.72 nM T64765 C7QXR1 44275844 Ki = 181.97 nM T64765 CIXC65 44275952 Ki = 6.166 nM T64765 CGA7Z0 44285139 Ki = 87 nM T64765 CL5YJ6 44294664 Ki = 152 nM T64765 C2WPH9 44294704 Ki = 28 nM T64765 CV08XD 44294847 Ki = 40 nM T64765 C3TMN4 44307705 Ki = 51.29 nM T64765 C45XRU 44307706 Ki = 758.58 nM T64765 C4JCB6 44307739 Ki = 43.65 nM T64765 CPOW71 44307766 Ki = 213.8 nM T64765 C1OS0D 44307778 Ki = 389.05 nM T64765 CT63YZ 44307779 Ki = 1.7 nM T64765 CCHI95 44307789 Ki < 1000 nM T64765 CUT1K7 44307791 Ki = 724.44 nM T64765 C4I0HR 44307802 Ki < 1000 nM T64765 CLI76H 44307804 Ki < 1000 nM T64765 CQF74O 44307839 Ki = 46.77 nM T64765 CAS52E 44307890 Ki < 1000 nM T64765 CS65LJ 44307891 Ki = 87.1 nM T64765 CH2XG4 44307899 Ki < 1000 nM T64765 C72PSH 44307904 Ki = 954.99 nM T64765 CWRL89 44307915 Ki = 251.19 nM T64765 CLHA64 44307916 Ki = 436.52 nM T64765 CN5V7T 44308031 Ki = 1000 nM T64765 C7YSB3 44308092 Ki = 44.67 nM T64765 CWK0X7 44308110 Ki = 158.49 nM T64765 CZ78OC 44308112 Ki = 53.7 nM T64765 CNK8I4 44308113 Ki = 158.49 nM T64765 CJ5AV7 44322449 Ki = 570 nM T64765 CEH42A 44322540 Ki = 65 nM T64765 COB0I5 44322550 Ki = 650 nM T64765 CY29GR 44322589 Ki = 190 nM T64765 C4BLC5 44335225 Ki = 15.14 nM T64765 C1TL7P 44335238 Ki = 2.138 nM T64765 C51LMP 44335336 Ki = 199.53 nM T64765 CCI26P 44335384 Ki = 7.079 nM T64765 CNF4S6 44335387 Ki = 1000 nM T64765 C2ZN6D 44335405 Ki = 117.49 nM T64765 C04MTD 44335456 Ki = 123.03 nM T64765 CO0GR9 44335463 Ki = 1000 nM T64765 CMD1U0 44335483 Ki = 30.2 nM T64765 C12MNS 44335558 Ki = 13.8 nM T64765 CJX50C 44335559 Ki = 1.698 nM T64765 CN9JI6 44335571 Ki = 36.31 nM T64765 CFLQ98 44340628 Ki = 4000 nM T64765 C07LOA 44341076 Ki = 4800 nM T64765 CT5W9X 44351678 Ki = 3.89 nM T64765 C6F5DP 44352445 Ki = 16 nM T64765 C4DK3A 44352460 Ki = 14 nM T64765 CS0E2H 44367567 EC50 = 2.089 nM T64765 CS2J8O 44367568 EC50 = 0.389 nM T64765 CKG9B4 44370611 Ki = 49 nM T64765 CNL6W8 44373673 Ki = 88 nM T64765 C6VON7 44373679 Ki = 18 nM T64765 CGFC57 44373680 Ki = 13 nM T64765 CL3W7O 44373686 Ki = 49 nM T64765 CT06KP 44373692 Ki = 85 nM T64765 C5R2SA 44373693 Ki = 160 nM T64765 C46HCQ 44373704 Ki = 36 nM T64765 CNI9Z6 44373706 Ki = 86 nM T64765 CFB17R 44373711 Ki = 43 nM T64765 C17YQC 44373712 Ki = 28 nM T64765 CET05N 44373720 Ki = 170 nM T64765 CE8Y7V 44373726 Ki = 130 nM T64765 CP6SJ4 44373727 Ki = 79 nM T64765 C7R3QK 44373749 Ki = 92 nM T64765 CU0KS5 44373750 Ki = 11 nM T64765 CM5V4X 44373760 Ki = 170 nM T64765 CL0UC3 44373762 Ki = 23 nM T64765 CY1Q9W 44373766 Ki = 16 nM T64765 C62SRU 44373776 Ki = 230 nM T64765 CLW1V5 44373784 Ki = 65 nM T64765 CK4C0J 44373785 Ki = 87 nM T64765 CK23QJ 44373786 Ki = 200 nM T64765 C19UVF 44373795 Ki = 110 nM T64765 C5PW9U 44373797 Ki = 8.6 nM T64765 CGCQ62 44373798 Ki = 17 nM T64765 CYJ72I 44373799 Ki = 18 nM T64765 CUCT36 44373835 Ki = 40 nM T64765 CH6WV5 44373843 Ki = 190 nM T64765 C71XFA 44373845 Ki = 42 nM T64765 C4P7LI 44373846 Ki = 29 nM T64765 C2VK6E 44373847 Ki = 27 nM T64765 CHB5F9 44373853 Ki = 85 nM T64765 CSEA06 44373855 Ki = 64 nM T64765 COB82T 44373858 Ki = 46 nM T64765 CBQ78F 44373859 Ki = 240 nM T64765 CH1D6T 44373867 Ki = 34 nM T64765 C8OJP4 44373870 Ki = 40 nM T64765 CA2L5O 44373873 Ki = 74 nM T64765 CT4P7F 44373874 Ki = 36 nM T64765 CG89XO 44373877 Ki = 80 nM T64765 CM59QC 44373878 Ki = 9.8 nM T64765 C73XLS 44373884 Ki = 520 nM T64765 C40LWD 44373892 Ki = 17 nM T64765 CZU2W6 44373893 Ki = 13 nM T64765 C3Z7IG 44373894 Ki = 43 nM T64765 CBA12O 44373898 Ki = 240 nM T64765 CUG8Z3 44373899 Ki = 26 nM T64765 CF5H0S 44373903 Ki = 40 nM T64765 CW9UK5 44373905 Ki = 8.6 nM T64765 CW4A9Q 44373912 Ki = 20 nM T64765 C12MLR 44373914 Ki = 14 nM T64765 C0Z4MG 44373915 Ki = 560 nM T64765 CT9UW6 44373917 Ki = 24 nM T64765 CCF75A 44373925 Ki = 39 nM T64765 CO0V1Z 44373930 Ki = 47 nM T64765 CB0X6G 44373931 Ki = 18 nM T64765 CBG07X 44373932 Ki = 140 nM T64765 CU6WL8 44373933 Ki = 15 nM T64765 CUTV25 44373934 Ki = 21 nM T64765 CA0EW2 44373941 Ki = 56 nM T64765 C7Q8YE 44373961 Ki = 110 nM T64765 CB9UT7 44373970 Ki = 34 nM T64765 CWCZ96 44373971 Ki = 54 nM T64765 C4UT0L 44373975 Ki = 8.6 nM T64765 CWP8H1 44374044 Ki = 13 nM T64765 CX0OM7 44374045 Ki = 37 nM T64765 C7GDZ5 44374046 Ki = 130 nM T64765 CMRD92 44374063 Ki = 49 nM T64765 CRC5G3 44374070 Ki = 100 nM T64765 CMH6V5 44374082 Ki = 75 nM T64765 CX16WJ 44374083 Ki = 92 nM T64765 C7I6MZ 44374097 Ki = 70 nM T64765 CZ9V8G 44374105 Ki = 15 nM T64765 CDQ6R1 44374106 Ki = 24 nM T64765 C9AU3H 44374107 Ki = 140 nM T64765 C87KSL 44374109 Ki = 40 nM T64765 C8OKT7 44374123 Ki = 19 nM T64765 CQTR45 44374124 Ki = 9.3 nM T64765 CYH60O 44374137 Ki = 16 nM T64765 CWM1V4 44374143 Ki = 110 nM T64765 CB6QC8 44374148 Ki = 31 nM T64765 CS7DA2 44374156 Ki = 98 nM T64765 C8BR9Y 44374157 Ki = 100 nM T64765 CYIA95 44374158 Ki = 68 nM T64765 CZ6V8G 44374162 Ki = 15 nM T64765 C8UEW3 44374165 Ki = 120 nM T64765 CN84FV 44374231 Ki = 31 nM T64765 C4G8HL 44374253 Ki = 12 nM T64765 C8TVJ2 44374254 Ki = 210 nM T64765 C9LTB6 44374276 Ki = 14 nM T64765 CW37NB 44374378 Ki = 20 nM T64765 CI70JD 44374379 Ki = 9.5 nM T64765 CCL93B 44374396 Ki = 35 nM T64765 CNS57W 44374397 Ki = 7.5 nM T64765 C3PS4N 44374398 Ki = 170 nM T64765 CN62CP 44374399 Ki = 520 nM T64765 CJ0H1Z 44374441 Ki = 0.7 nM T64765 CXL65I 44374451 Ki = 5.1 nM T64765 CH4W8B 44374493 Ki = 0.5495 nM T64765 C0HJK7 44374555 Ki = 1.9 nM T64765 C4P3NO 44374578 Ki = 316.23 nM T64765 CLO3V5 44374695 Ki = 5.888 nM T64765 CP4RS0 44374751 Ki = 36 nM T64765 C59JWF 44374769 Ki = 5.6 nM T64765 CI9JB8 44385102 Ki = 1.1 nM T64765 CP4S5Y 44385157 Ki = 18 nM T64765 C1OL7T 44386214 Ki = 19 nM T64765 CY51NG 44395308 Ki = 2511.89 nM T64765 CUW8B3 44395314 EC50 = 1000 nM T64765 CHU6B8 44395335 EC50 = 3162.28 nM T64765 C9QSE7 44395364 EC50 = 1000 nM T64765 C53DOL 44407694 Ki = 8 nM T64765 C6CJ0K 44407728 Ki = 36 nM T64765 C7MU4O 44407729 Ki = 18 nM T64765 C0RH8D 44407809 Ki = 40 nM T64765 CWV3C9 44407928 Ki = 14 nM T64765 CEP8K7 44409909 Ki = 351 nM T64765 CCZ4N6 44409953 Ki = 178 nM T64765 C8O7FH 44409954 Ki = 31 nM T64765 C49TLG 44409955 Ki = 31 nM T64765 C1WU9K 44409959 Ki = 170 nM T64765 C97OWX 44409960 Ki = 11 nM T64765 CI4NM3 44411554 Ki > 150 nM T64765 C0BLI1 44411604 Ki = 14 nM T64765 CFMT69 44411608 Ki = 11 nM T64765 CLMD61 44411609 Ki = 5 nM T64765 C62RDP 44411615 Ki > 150 nM T64765 CTM46Z 44411619 Ki = 15 nM T64765 CQCD08 44411624 Ki = 22 nM T64765 CPE46Q 44411625 Ki = 46 nM T64765 CH3W7I 44411629 Ki = 7 nM T64765 CNXO69 44411921 Ki = 12 nM T64765 CF3SN2 44411922 Ki = 5 nM T64765 CRZ57N 44411927 Ki = 4 nM T64765 CSRK30 44411928 Ki = 7 nM T64765 CR4CY6 44412593 Ki = 0.6 nM T64765 C8BQS2 44412594 Ki = 0.35 nM T64765 CX87JP 44412616 Ki = 0.53 nM T64765 CD03TZ 44412617 Ki = 7.4 nM T64765 C6MVQ2 44412634 Ki = 2.1 nM T64765 C0S4HM 44412635 Ki = 8.1 nM T64765 CRB98T 44412649 Ki = 154 nM T64765 C8OEI2 44412650 Ki = 0.17 nM T64765 CDOQ83 44412667 Ki = 4.9 nM T64765 CN1VJ2 44412668 Ki = 23.8 nM T64765 CGV0C9 44412695 Ki = 95 nM T64765 C6HV1L 44412696 Ki > 300 nM T64765 C8WYV5 44412697 Ki > 300 nM T64765 C0FR5P 44412698 Ki > 300 nM T64765 CN6UQ2 44412699 Ki = 19.4 nM T64765 CJOS82 44412714 Ki = 59 nM T64765 C5RU1E 44412715 Ki > 300 nM T64765 CC8J3R 44412716 Ki > 300 nM T64765 CTE21L 44412733 Ki > 300 nM T64765 CYCF41 44412745 Ki = 84 nM T64765 CUH45T 44412760 Ki = 15.4 nM T64765 CQZ40L 44412761 Ki > 300 nM T64765 C6YED7 44412777 Ki > 300 nM T64765 C35BVA 44412778 Ki > 300 nM T64765 C02BVG 44412800 Ki = 1.01 nM T64765 C42LIZ 44414343 Ki = 46.77 nM T64765 C8UV1I 44414367 Ki = 1412.54 nM T64765 CK0Q1G 44414369 Ki = 6.31 nM T64765 CXK6C4 44414370 Ki = 1.698 nM T64765 CZH9M7 44414393 Ki = 1.175 nM T64765 CKEM26 44414417 Ki = 562.34 nM T64765 C9X2SV 44414433 Ki = 758.58 nM T64765 CXW0G2 44414480 Ki = 6.166 nM T64765 CC51VO 44414495 Ki = 398.11 nM T64765 CH7D4C 44414498 Ki = 37.15 nM T64765 CCW06N 44414519 Ki = 12.3 nM T64765 CVF74L 44418464 Ki = 281 nM T64765 C2S3EF 44418465 Ki = 37 nM T64765 C04THX 44418471 Ki = 94 nM T64765 CS6PZ7 44418472 Ki = 59 nM T64765 C9XDL2 44418473 Ki = 45 nM T64765 C49MQF 44418477 Ki = 23 nM T64765 CQ2D0O 44418482 Ki = 25 nM T64765 CPTD84 44418489 Ki = 14 nM T64765 CX09NV 44418490 Ki = 47 nM T64765 C68QUP 44418491 Ki = 73 nM T64765 CR35FG 44418496 Ki = 11.2 nM T64765 CV5PD9 44418497 Ki = 16 nM T64765 CU8B2E 44418498 Ki = 86 nM T64765 C6YX3F 44418499 Ki = 27 nM T64765 CN8X7R 44418504 Ki = 13.4 nM T64765 C10MOB 44418505 Ki = 3.7 nM T64765 CUH08F 44418511 Ki = 162 nM T64765 CAUW81 44418512 Ki = 165 nM T64765 C9EXM4 44418519 Ki = 121 nM T64765 C4RIA6 44418520 Ki = 87 nM T64765 CNE92B 44418526 Ki = 196 nM T64765 CM42CY 44418527 Ki = 295 nM T64765 CS2DU7 44418528 Ki = 188 nM T64765 CZ8K5R 44418534 Ki = 117 nM T64765 CUO0K4 44418535 Ki = 78 nM T64765 CM4W3U 44418536 Ki = 109 nM T64765 CT67AU 44418541 Ki = 34 nM T64765 CMU5P3 44418542 Ki = 47 nM T64765 C5VQ3A 44418548 Ki = 458 nM T64765 C1VA7G 44418549 Ki = 226 nM T64765 CVN7E2 44418550 Ki = 52 nM T64765 CN3EH8 44418558 Ki = 29 nM T64765 CJ6R9G 44418559 Ki = 30 nM T64765 C90KAM 44418565 Ki = 44 nM T64765 CPD82E 44418566 Ki = 40 nM T64765 CL6WE1 44418567 Ki = 38 nM T64765 CVFN23 44418574 Ki = 34 nM T64765 C0WFA9 44418575 Ki = 15 nM T64765 C5EU2J 44418576 Ki = 20 nM T64765 CGD45W 44425550 Ki = 18 nM T64765 C0SIH8 44425551 Ki = 1021 nM T64765 CT1DN3 44425552 Ki = 150 nM T64765 C0U7YR 44425553 Ki = 88 nM T64765 CU7N0Z 44425554 Ki = 135 nM T64765 CWD9M2 44425555 Ki = 2.4 nM T64765 C6ANE3 44425557 Ki = 47 nM T64765 CXST62 44425559 Ki = 1100 nM T64765 C0DX4K 44425560 Ki = 1810 nM T64765 C7ZY6M 44425561 Ki = 1393 nM T64765 C1ON3Q 44425562 Ki = 12 nM T64765 C2JOU8 44430356 Ki = 69 nM T64765 C90VJB 44430358 Ki = 9.5 nM T64765 CBOP25 44430359 Ki = 47 nM T64765 CD0E3S 44430363 Ki = 38 nM T64765 C01VKH 44430365 Ki = 7.4 nM T64765 C4T7KP 44430367 Ki = 12 nM T64765 CZB0W3 44430368 Ki = 9.7 nM T64765 C1Z6WS 44430371 Ki = 30 nM T64765 C4KA7J 44430373 Ki = 1108 nM T64765 CDP69G 44430375 Ki = 144 nM T64765 CR1IT7 44430379 Ki = 268 nM T64765 CU1F0L 44430380 Ki = 3.3 nM T64765 C07PLN 44430381 Ki = 1440 nM T64765 CZJ2W5 44434147 Ki = 5.4 nM T64765 CN8A3O 44434150 Ki = 13 nM T64765 CF42IC 44434165 Ki = 6.1 nM T64765 CY79ZO 44434236 Ki = 4 nM T64765 CCS8D1 44434250 Ki = 9.7 nM T64765 C1I2BU 44437495 Ki = 5150 nM T64765 CS9UQ1 44437496 Ki > 1000 nM T64765 C4SV8L 44437497 Ki > 1000 nM T64765 CO8DT9 44437498 Ki > 1000 nM T64765 C9R8WN 44437499 Ki = 1420 nM T64765 C3ZDU4 44437500 Ki = 581 nM T64765 CP36JI 44437501 Ki = 9990 nM T64765 CCMV89 44437514 Ki = 2800 nM T64765 CO20QU 44437515 Ki > 1000 nM T64765 CW09ML 44437517 Ki = 6510 nM T64765 CE5OX7 44437518 Ki > 1000 nM T64765 CXH06Q 44437519 Ki = 853 nM T64765 CYK2O7 44437520 Ki > 1000 nM T64765 CAV9L2 44437522 Ki = 2080 nM T64765 C4HZX3 44437523 Ki = 1010 nM T64765 CXBE83 44437524 Ki = 1050 nM T64765 C4X0AD 44437525 Ki = 1630 nM T64765 CPLN85 44437526 Ki = 1130 nM T64765 CTKX20 44437528 Ki = 548 nM T64765 CE08HO 44437541 Ki = 779 nM T64765 C7VBE4 44437542 Ki = 629 nM T64765 CV6S2Q 44437544 Ki = 1310 nM T64765 CYC56F 44437547 Ki = 807 nM T64765 CPDS73 44437553 Ki > 1000 nM T64765 CZ9L4F 44437555 Ki = 9260 nM T64765 C1AU2N 44437557 Ki = 6680 nM T64765 C0IQ8W 44437609 Ki > 1000 nM T64765 CBG34A 44437612 Ki = 899 nM T64765 CC1L2V 44437614 Ki = 2140 nM T64765 CJQ1X5 44437620 Ki = 8800 nM T64765 CVJ05I 44438666 Ki = 7 nM T64765 C5Q3LJ 44438903 Ki = 0.9 nM T64765 C6U4CQ 44438905 Ki = 2 nM T64765 CG1CI3 44438906 Ki = 4 nM T64765 CWM1C9 44438907 Ki = 2 nM T64765 C08WVG 44438908 Ki = 2.2 nM T64765 CRX6J5 44438910 Ki = 1.2 nM T64765 C1NBD8 44438911 Ki = 2.3 nM T64765 CWN70H 44438913 Ki = 1.7 nM T64765 CF6PY1 44438915 Ki = 1.2 nM T64765 C4M6FA 44438918 Ki = 1.3 nM T64765 C86YHM 44438919 Ki = 4.7 nM T64765 C2WK5Z 44438926 Ki = 2 nM T64765 CB3PK5 44438927 Ki = 4 nM T64765 C5RSG7 44438935 Ki = 2.5 nM T64765 CAH1X0 44438939 Ki = 0.7 nM T64765 C31BWH 44438944 Ki = 1.7 nM T64765 C3Q8OY 44438945 Ki = 1.3 nM T64765 CRTK53 44438946 Ki = 1.7 nM T64765 CH4U2Z 44438947 Ki = 0.7 nM T64765 CT18FP 44438948 Ki = 3.7 nM T64765 C3GB8R 44438949 Ki = 1.6 nM T64765 CF9R8D 44439854 Ki = 7.3 nM T64765 CS1LB8 44439855 Ki = 5.6 nM T64765 CDX7C5 44439856 Ki = 3.3 nM T64765 CY5J2W 44439857 Ki = 18 nM T64765 C10ZYB 44439858 Ki = 11 nM T64765 C3IJ7Y 44439859 Ki = 3.5 nM T64765 CHKE50 44439860 Ki = 8.3 nM T64765 CR1FY4 44439861 Ki = 46 nM T64765 CP9B4A 44439862 Ki = 6.9 nM T64765 C50ZDW 44439863 Ki = 5.6 nM T64765 C9HP5V 44440807 Ki = 0.22 nM T64765 CH70BJ 44440809 Ki = 3.31 nM T64765 CU9Z4B 44440856 Ki = 19.95 nM T64765 CSRF79 44440857 Ki = 8.71 nM T64765 C0ZG5V 44440868 Ki = 1.09 nM T64765 CMH69J 44440872 Ki = 10.47 nM T64765 CZK1U5 44441058 Ki = 5.3 nM T64765 CF8K5H 44441067 Ki = 0.8 nM T64765 C6VC8I 44441070 Ki = 1.6 nM T64765 CFCO97 44441071 Ki = 0.8 nM T64765 C1O9VZ 44441073 Ki = 2.7 nM T64765 CI43TX 44441077 Ki = 1 nM T64765 CZOU36 44441079 Ki = 3 nM T64765 CV0UI9 44441083 Ki = 3 nM T64765 CITP46 44441084 Ki = 3.7 nM T64765 CX7N0I 44441085 Ki = 3.3 nM T64765 C69RCY 44441088 Ki = 4 nM T64765 CC0A8B 44441089 Ki = 2 nM T64765 CJ7Z3F 44447974 Ki = 83 nM T64765 CC9P0H 44447975 Ki = 36 nM T64765 C2PV7W 44447976 Ki = 24 nM T64765 CF30GS 44447977 Ki = 6.6 nM T64765 CHBE43 44447978 Ki = 16 nM T64765 CWS5M2 44447979 Ki = 2.4 nM T64765 CP1BA6 44447980 Ki = 61 nM T64765 CFGQ89 44447981 Ki = 56 nM T64765 CIM2S3 44447985 Ki = 0.38 nM T64765 CYRO07 44447986 Ki = 1.3 nM T64765 CL40DS 44447987 Ki = 0.47 nM T64765 C76BJN 44447988 Ki = 0.34 nM T64765 CXP2J1 44451644 Ki = 0.6761 nM T64765 CAV5I8 44454614 Ki = 0.9 nM T64765 CZL97F 44455426 Ki > 10000 nM T64765 CC09EJ 44455512 Ki = 1.1 nM T64765 C16SFL 44455822 Ki = 0.9 nM T64765 CB8AN0 44455850 Ki = 0.5 nM T64765 CEY02T 44455851 Ki = 1 nM T64765 C84UEC 44455913 Ki = 1.6 nM T64765 CQ34CF 44455918 Ki = 1.3 nM T64765 C3F4GB 44455919 Ki > 330 nM T64765 C1B8XT 44455947 Ki = 3.5 nM T64765 CJBQ07 44455987 Ki = 28 nM T64765 C16EDN 44455990 Ki = 26 nM T64765 CQT0R1 44455991 Ki = 15 nM T64765 C1NQY6 44456024 Ki = 100 nM T64765 CT1KJ3 44456052 Ki = 132 nM T64765 C35NGB 44456058 Ki = 18 nM T64765 CT70DM 44456231 Ki = 20 nM T64765 COW12C 44456292 Ki = 11 nM T64765 C08MBY 44456312 Ki = 2.4 nM T64765 C1WQF2 44456333 Ki = 10 nM T64765 C12XGE 44456400 Ki > 10000 nM T64765 CEUV85 44456404 Ki = 43 nM T64765 C1E0YI 44456405 Ki = 6 nM T64765 C9XS5D 44456406 Ki > 360 nM T64765 CVZ5N1 44456407 Ki > 360 nM T64765 C8XYE0 44456408 Ki = 110 nM T64765 C1ZXT2 44456409 Ki = 34 nM T64765 CW0P9X 44456446 Ki = 17 nM T64765 CS5BD4 44456449 Ki = 33 nM T64765 CN4SP3 44456450 Ki = 34 nM T64765 CP05GX 44456497 Ki = 300 nM T64765 CQ0WM7 44469273 IC50 > 5000 nM T64765 CK10AW 44478385 Ki = 524.81 nM T64765 C7GMD8 44480959 EC50 = 251.19 nM T64765 CDC6Z1 44517827 Ki = 30 nM T64765 C14SNF 44539764 Ki = 10 nM T64765 CI75BA 44539765 Ki = 134 nM T64765 CD2JT1 44539766 Ki = 167 nM T64765 CF2P3I 44539768 Ki = 16 nM T64765 C8J3XG 44539769 Ki = 17 nM T64765 CBF9E1 44539868 Ki = 31 nM T64765 C8YN1J 44539869 Ki = 8 nM T64765 C7G0NQ 44539870 Ki = 5 nM T64765 CAW1H3 44539969 Ki = 83 nM T64765 CMW56J 44539973 EC50 = 2 nM T64765 CF3RX5 44539976 Ki = 34 nM T64765 C0RA9E 44540072 EC50 = 2.1 nM T64765 C8W3ZH 44540074 Ki = 47 nM T64765 CJ8U5S 44546761 Ki = 1760 nM T64765 CIUF42 44546762 Ki = 130 nM T64765 CV21YF 44546763 Ki = 2130 nM T64765 C5NEC7 44546913 Ki = 1650 nM T64765 CZ8E9W 44546914 Ki = 1360 nM T64765 C1XPV7 44546915 Ki = 150 nM T64765 CUS9L0 44546916 Ki = 1550 nM T64765 C7EZ4V 44546917 Ki = 1520 nM T64765 CM7YC2 44548785 Ki = 270 nM T64765 CQ0JU2 44548786 Ki = 430 nM T64765 C7OL2Z 44548787 Ki = 120 nM T64765 C9CFM7 44548788 Ki = 250 nM T64765 C0XL5R 44548789 Ki = 210 nM T64765 CIO48H 44548938 Ki = 440 nM T64765 C0DOR3 44549084 Ki = 1610 nM T64765 CP06NU 44549085 Ki = 80 nM T64765 C5QL9B 44549086 Ki = 670 nM T64765 C5FGS2 44549087 Ki = 1250 nM T64765 C5HY0K 44549088 Ki = 190 nM T64765 C9RH4J 44549089 Ki = 1610 nM T64765 C0NVX8 44549090 Ki = 1330 nM T64765 C1H3CM 44560976 Ki = 2 nM T64765 CS6W4N 44562525 Ki = 38 nM T64765 CT9S4L 44563063 Ki = 0.5 nM T64765 CDTB89 44563137 Ki = 0.2188 nM T64765 C1VZ4R 44563682 Ki = 560 nM T64765 C8MC0F 44563686 Ki = 393 nM T64765 CZC96U 44563687 Ki = 235 nM T64765 C7C8TE 44563697 Ki = 132 nM T64765 CHD29R 44563698 Ki > 10000 nM T64765 CXF02W 44563699 Ki = 164 nM T64765 CP03NM 44563700 Ki = 300 nM T64765 CJ2V7G 44563701 Ki = 176 nM T64765 CB3HT4 44563702 Ki = 165 nM T64765 CVA67X 44568347 Ki = 960 nM T64765 C2BEA0 44570656 Ki = 18 nM T64765 CNE4V5 44571276 Ki = 70 nM T64765 C96PAU 44571277 Ki = 1 nM T64765 C3HFM6 44571278 Ki = 24 nM T64765 CRO79N 44571343 Ki = 71 nM T64765 CML90U 44578389 Ki = 1.094 nM T64765 CGBH19 44578605 Ki = 57 nM T64765 C38CNA 44578637 EC50 = 21 nM T64765 C9CZ3D 44579387 IC50 = 110 nM T64765 CDR85P 44579388 IC50 = 343 nM T64765 C42JUT 44579389 IC50 = 893 nM T64765 CJNE08 44579427 IC50 = 680 nM T64765 C70WKN 44579428 IC50 = 393 nM T64765 CONH50 44579429 IC50 = 237 nM T64765 C7KPA3 44579430 IC50 = 530 nM T64765 C6MI8V 44579431 IC50 = 98 nM T64765 CP15YC 44579472 IC50 = 267 nM T64765 CJ54WS 44579473 IC50 > 1000 nM T64765 CC0ER4 44579474 IC50 = 506 nM T64765 CD42OL 44579475 IC50 > 1000 nM T64765 CA4S5V 44579476 IC50 = 297 nM T64765 C6NX9B 44579547 IC50 = 160 nM T64765 C8ZI4B 44579548 IC50 > 1000 nM T64765 CL26TJ 44579549 IC50 = 783 nM T64765 CZ75OF 44579550 IC50 > 1000 nM T64765 C7URO6 44579551 IC50 = 560 nM T64765 CDI14W 44579606 IC50 = 380 nM T64765 CIGA58 44579607 IC50 = 68 nM T64765 CVN4D6 44580259 Ki = 11 nM T64765 C4RNV0 44580338 Ki = 4.8 nM T64765 C6KTZ4 44580339 Ki = 3.6 nM T64765 CE87QS 44580381 Ki = 107 nM T64765 C3KXZ2 44580382 Ki = 713 nM T64765 C9B2LH 44580383 Ki = 16 nM T64765 CLH08J 44580429 Ki = 20 nM T64765 C2VQG9 44580430 Ki = 11 nM T64765 C70IOM 44580431 Ki = 101 nM T64765 C78CMV 44580432 Ki = 8.7 nM T64765 CW74NK 44580468 Ki = 8 nM T64765 CEQ74T 44580469 Ki = 2.6 nM T64765 C46CQG 44580470 Ki = 15 nM T64765 CO1H2B 44581055 Ki = 2100 nM T64765 C8B4OK 44581056 Ki = 165 nM T64765 CA5Z3U 44581057 Ki = 106 nM T64765 C7QM8L 44581058 Ki = 49 nM T64765 C54QPF 44581059 Ki = 18 nM T64765 CFC05J 44581060 Ki = 3.6 nM T64765 COF5D0 44581076 Ki = 566 nM T64765 C6RF8I 44581077 Ki = 102 nM T64765 C7MGZ9 44581078 Ki = 37 nM T64765 CV9H7B 44581095 Ki = 7100 nM T64765 C5ND3T 44581096 Ki > 10000 nM T64765 C70HRP 44581097 Ki = 5300 nM T64765 CEKR10 44581098 Ki = 2.2 nM T64765 CJGC41 44581099 Ki = 2.5 nM T64765 CSNC81 44581100 Ki = 31 nM T64765 CJ7UB6 44582618 Ki = 12.5 nM T64765 CI2OT0 44582619 Ki = 7.2 nM T64765 CQY7X5 44582670 Ki = 27.3 nM T64765 CNJW59 44582671 Ki = 49 nM T64765 C8NRM2 44582672 Ki = 18.6 nM T64765 C6T9AI 44582673 Ki = 3.2 nM T64765 C03AIU 44582674 Ki = 3.5 nM T64765 CRCH48 44582675 Ki > 10000 nM T64765 CEJ4R8 44582676 Ki > 10000 nM T64765 C5QB4K 44582678 Ki > 10000 nM T64765 C7NR1M 44582701 Ki = 12.8 nM T64765 CSN1W3 44582702 Ki = 51 nM T64765 CQ2N8E 44582703 Ki = 7.7 nM T64765 CZE73M 44582704 Ki = 2.4 nM T64765 C01RCI 44582705 Ki = 9033 nM T64765 C80BWF 44588111 Ki = 2.818 nM T64765 CZ9D6V 44588146 Ki = 9.333 nM T64765 CA6QG0 44588178 Ki = 2.754 nM T64765 CK0JH4 44588213 Ki = 0.871 nM T64765 C6N5CA 44588214 Ki = 19.5 nM T64765 C8ZO5X 44588215 Ki = 75.86 nM T64765 C5AIM1 44588216 Ki = 2.188 nM T64765 C0B1MX 44588217 Ki = 1.95 nM T64765 CA17JI 44588248 Ki = 1.738 nM T64765 C3CU0X 44588249 Ki = 2.399 nM T64765 C42TLD 44588250 Ki = 6.761 nM T64765 C49BUZ 44588277 Ki = 5.129 nM T64765 CMO28B 44588278 Ki = 16.6 nM T64765 CWX3R0 44588348 Ki = 251.19 nM T64765 CO3FH8 44588349 Ki = 8.511 nM T64765 CSA15P 44588350 Ki = 3.89 nM T64765 CP6ZA9 44591012 Ki = 4.9 nM T64765 CU37BO 44591098 Ki = 3.5 nM T64765 CU48CL 44591099 Ki = 0.25 nM T64765 C7H9SE 44591134 Ki = 1.21 nM T64765 C6RLW0 44591135 Ki = 1.54 nM T64765 C8CUV1 44592066 Ki = 0.09333 nM T64765 CA6QH9 44592095 Ki > 1000 nM T64765 CN4A0M 44592098 Ki = 0.28 nM T64765 COX6H1 44592126 Ki = 0.28 nM T64765 CL6OI4 44592127 Ki = 0.26 nM T64765 CNV21B 44592128 Ki = 0.31 nM T64765 CMG26R 44592129 Ki = 0.99 nM T64765 COJE45 44592130 Ki = 0.24 nM T64765 CI8OV6 44592131 Ki = 0.2 nM T64765 CK13NZ 44592165 Ki = 0.068 nM T64765 C69VHJ 44592166 Ki = 0.8318 nM T64765 C6J2NP 44598901 Ki = 840 nM T64765 CM2UG7 44598902 Ki = 1.6 nM T64765 CZU8H2 44598903 Ki = 5.4 nM T64765 CP7XQ0 44598904 Ki = 6 nM T64765 C8WFL9 44598905 Ki = 2.7 nM T64765 CQC79I 44598906 Ki = 3.7 nM T64765 C48ZOE 44599076 Ki = 600 nM T64765 C9J1WH 44599235 Ki = 2.2 nM T64765 C5ZAY2 44599236 Ki = 13 nM T64765 CNPO87 44599397 Ki = 1970 nM T64765 C4VPI7 44599399 Ki = 200 nM T64765 C2UI0Z 44599400 Ki = 11 nM T64765 C1CZX3 44600840 Ki = 2.8 nM T64765 CQ6EU0 44600841 Ki = 1.3 nM T64765 CM7D9V 44600842 Ki = 5 nM T64765 CA8Z2U 44600843 Ki = 5.2 nM T64765 C2DJ5K 44600844 Ki = 4.1 nM T64765 CTR34Y 44600845 Ki = 4.7 nM T64765 CVJG25 44600846 Ki = 4.1 nM T64765 CR2JS4 44600994 Ki = 37 nM T64765 CJHP46 44601157 Ki = 54 nM T64765 CR8FY2 44601323 Ki = 7.5 nM T64765 C4ID9A 44602971 Ki = 2 nM T64765 C7I4EY 44603096 Ki = 2 nM T64765 C0WVZ1 44622338 Ki = 36 nM T64765 CL26YD 44622339 Ki = 1 nM T64765 CA7EQ2 44622340 Ki = 2 nM T64765 C23ORN 44622341 Ki = 1 nM T64765 C2JIX6 44622342 Ki = 1 nM T64765 CNI29G 44622416 Ki = 2 nM T64765 C9KUD5 44622417 Ki = 2 nM T64765 C4Q7JB 44622418 Ki = 2 nM T64765 C12SGH 44622499 Ki = 15 nM T64765 C3Q7BW 44816514 Ki = 7 nM T64765 CK5CO3 44816517 Ki = 11 nM T64765 C85DWU 44816692 Ki = 4 nM T64765 CT58XF 44816866 Ki = 7 nM T64765 CYXD79 45257131 Ki = 446.68 nM T64765 C07WHQ 45257132 Ki = 512.86 nM T64765 CY25IH 45257133 Ki = 346.74 nM T64765 C5ND1K 45263439 EC50 = 316.23 nM T64765 CLCM07 45266943 Ki = 26400 nM T64765 C6U9DR 45266945 Ki = 2290 nM T64765 CZNG94 45267022 Ki = 32500 nM T64765 C9U4VM 45267023 Ki = 310 nM T64765 CP63NC 45267051 Ki = 2110 nM T64765 CQH4L3 45267230 Ki = 7.943 nM T64765 C3X7CM 45267233 Ki = 7.943 nM T64765 C46QKW 45267237 Ki = 12.59 nM T64765 C3T5PI 45267459 Ki = 0.2 nM T64765 C2F9HZ 45267888 Ki = 2720 nM T64765 CED2I6 45267891 Ki = 537 nM T64765 C9CNJ8 45267892 Ki = 1100 nM T64765 CWL5Y3 45268093 Ki = 3.162 nM T64765 CEJ07N 45268095 Ki = 31.62 nM T64765 C0XAR6 45268283 IC50 = 3 nM T64765 C7V1WF 45268290 IC50 = 8.6 nM T64765 C9RCS2 45268299 IC50 = 0.4 nM T64765 CLF90U 45268300 Ki = 0.3 nM T64765 C2T0ZC 45268315 IC50 = 0.6 nM T64765 CO4CB9 45268759 Ki = 776 nM T64765 CUG4V7 45268970 Ki = 19.95 nM T64765 C53UBD 45269440 Ki = 62 nM T64765 CL2U8F 45269614 Ki = 17600 nM T64765 C6PA5C 45269622 Ki = 170 nM T64765 C2BDA9 45269627 Ki = 89.1 nM T64765 CF36SE 45269820 Ki = 7.943 nM T64765 C8C2AK 45270025 IC50 = 1.8 nM T64765 C2L8JN 45270044 IC50 = 0.39 nM T64765 COP3A7 45270277 Ki = 571 nM T64765 C5YUW8 45270644 Ki = 79.43 nM T64765 CUV67Q 45270855 IC50 = 5.9 nM T64765 C5UP2J 45270862 IC50 = 0.84 nM T64765 CEM4Z0 45270863 IC50 = 0.44 nM T64765 C9GK5C 45270870 IC50 = 0.34 nM T64765 C3LY0D 45271288 Ki = 61.66 nM T64765 C3O2FS 45271289 Ki = 15.85 nM T64765 C24QGO 45271464 Ki = 5.012 nM T64765 CC85BP 45271470 Ki = 6.31 nM T64765 CN4W1B 45271701 IC50 = 3.9 nM T64765 CW0JQ7 45271712 IC50 = 0.16 nM T64765 CAO92B 45271713 IC50 = 0.16 nM T64765 CVKI17 45271971 Ki = 36 nM T64765 C3C5TG 45271981 Ki = 234 nM T64765 CB29NU 45271982 Ki = 103 nM T64765 C2G6OU 45271991 Ki = 154 nM T64765 C0W5DO 45272163 Ki = 12900 nM T64765 CPU58M 45272172 Ki = 13500 nM T64765 CGV7P0 45272576 IC50 = 6.7 nM T64765 CR1F7A 45272583 IC50 = 0.6 nM T64765 C1TLM4 45272592 Ki = 0.8 nM T64765 CB5R3O 45272828 Ki = 30 nM T64765 C0GK4R 45273485 Ki = 0.6 nM T64765 CV8B6D 45273769 Ki = 2000 nM T64765 CMNA70 45358442 Ki > 630.96 nM T64765 CJN01K 45376015 Ki = 2.1 nM T64765 C6J3DG 45377353 Ki = 600.9 nM T64765 C7SYM5 45377639 Ki = 75 nM T64765 C96FQK 45377640 Ki = 12 nM T64765 C1RI6Z 45377641 Ki = 4.6 nM T64765 CC47NJ 45377915 Ki = 22.1 nM T64765 C6NG4K 45377916 Ki = 8.4 nM T64765 CX3K2N 45377917 Ki = 64.4 nM T64765 CD9EW7 45482497 Ki = 83.18 nM T64765 CE3P9Y 45482498 Ki = 56.23 nM T64765 C91UWI 45482679 Ki = 4 nM T64765 CP1YN5 45482680 Ki = 20 nM T64765 CR7Y5Z 45482682 Ki = 73 nM T64765 COI79T 45482683 Ki = 35 nM T64765 CV56HF 45482684 Ki = 10 nM T64765 C2C1XZ 45482685 Ki = 13 nM T64765 CA45ZR 45482686 Ki = 42 nM T64765 CGP38T 45482687 Ki = 133 nM T64765 CHV1Q5 45482688 Ki = 42 nM T64765 CUV0B2 45482692 Ki = 53 nM T64765 CK2G6S 45482693 Ki = 22 nM T64765 C9L4FG 45482694 Ki = 93 nM T64765 CEY8O1 45482699 Ki = 64 nM T64765 C2NM9W 45482703 Ki = 1700 nM T64765 C0SDI5 45482704 Ki = 141 nM T64765 C7W0DZ 45482705 Ki = 16 nM T64765 CP2ZT9 45482708 Ki = 28 nM T64765 CRL9I4 45482709 Ki = 104 nM T64765 C9UE0Y 45482713 Ki = 23 nM T64765 CH3S1P 45482714 Ki = 33 nM T64765 C8QJR2 45482726 Ki = 79 nM T64765 C3P5TG 45482727 Ki = 10 nM T64765 CZM43G 45482728 Ki = 8 nM T64765 C8IHQ4 45482743 Ki = 140 nM T64765 C89XKP 45482744 Ki = 59 nM T64765 CHQ4M5 45482745 Ki = 25 nM T64765 CJ3X8T 45482746 Ki = 25 nM T64765 C3NC6W 45482751 Ki = 16 nM T64765 CX9RG6 45482752 Ki = 66 nM T64765 C28XSF 45482753 Ki = 27 nM T64765 CW1T6S 45482755 Ki = 36 nM T64765 CZLA81 45482756 Ki = 35 nM T64765 CIH4Z3 45482757 Ki = 25 nM T64765 CLEQ10 45482761 Ki = 126 nM T64765 CSBL53 45482762 Ki = 46 nM T64765 C4EIV8 45482763 Ki = 17 nM T64765 CE0H4S 45482770 Ki = 44 nM T64765 C9DR7V 45482773 Ki = 80 nM T64765 C9ZDT6 45482774 Ki = 230 nM T64765 CLKA86 45482775 Ki = 35 nM T64765 C9W1NU 45482779 Ki = 125 nM T64765 CST3O8 45482780 Ki = 31 nM T64765 C2ED8W 45482783 Ki = 63 nM T64765 C3QU2C 45487384 IC50 > 5000 nM T64765 C5WRZ1 46182734 Ki = 103 nM T64765 C0T7YF 46194892 IC50 <= 50 nM T64765 C5KFD3 46212800 IC50 = 66 nM T64765 CB04XO 46212809 IC50 = 48 nM T64765 C6U0CX 46212866 IC50 = 11 nM T64765 CTZ46V 46220927 Ki = 19.8 nM T64765 CJI65Q 46220928 Ki = 63 nM T64765 CX18IP 46221142 Ki = 6.7 nM T64765 CBIU25 46221376 Ki = 129 nM T64765 C53NBG 46230561 Ki = 1200 nM T64765 CE28MP 46230600 Ki = 235 nM T64765 CQ1BF7 46230601 Ki = 23 nM T64765 CG8WQ0 46230602 Ki = 10 nM T64765 CY3FB2 46230635 Ki = 27 nM T64765 CJT03Q 46230636 Ki = 400 nM T64765 CBIS12 46230637 Ki = 4000 nM T64765 C8JXE5 46230691 Ki = 15 nM T64765 C1E0HI 46230692 Ki = 150 nM T64765 CYDL15 46230693 Ki = 130 nM T64765 CQDU07 46231335 Ki = 91 nM T64765 CU15OL 46235428 EC50 = 9000 nM T64765 CGAM07 46244628 Ki = 1200 nM T64765 CVED21 46244629 Ki = 4000 nM T64765 CZBY37 46244801 Ki = 657 nM T64765 CZG5R0 46244802 Ki = 253 nM T64765 C96YKR 46244804 Ki = 37 nM T64765 CN75IJ 46830167 EC50 = 1.862 nM T64765 CWRQ35 46861747 Ki = 1.8 nM T64765 CC5IO9 46861756 Ki = 1.5 nM T64765 C4VS0Q 46866435 IC50 = 3500 nM T64765 C18PID 46866437 Ki = 4.26 nM T64765 CG48EX 46866438 IC50 = 490 nM T64765 CCR8B5 46866439 IC50 = 790 nM T64765 CZ8VS6 46879683 Ki = 13 nM T64765 CW84GY 46879725 Ki = 28 nM T64765 CZ57FW 46879726 Ki = 43 nM T64765 C59ABH 46880384 Ki = 1.995 nM T64765 CYV93A 46880385 Ki = 7.943 nM T64765 CF83YX 46880387 Ki = 10 nM T64765 CIQ9Z5 46880446 Ki = 7.943 nM T64765 CG3D5X 46880447 Ki = 5.012 nM T64765 C9SFW5 46880448 Ki = 50.12 nM T64765 CPDQ25 46881855 Ki = 223.87 nM T64765 C15KEH 46883819 Ki = 86 nM T64765 C3J5IG 46883820 Ki = 67 nM T64765 C4TPV9 46883821 Ki > 1000 nM T64765 CC1NR9 46883822 Ki > 1000 nM T64765 C2Z7XO 46883875 Ki > 1000 nM T64765 CGKP83 46883876 Ki = 16 nM T64765 C3QL6X 46883877 Ki = 624 nM T64765 CJ39QM 46883878 Ki = 3 nM T64765 CXIM81 46883917 Ki = 49 nM T64765 C3OBL5 46883918 Ki = 2 nM T64765 CR6FO1 46883919 Ki = 10 nM T64765 CYC64I 46884402 Ki = 36 nM T64765 CN23CE 46884403 Ki = 191 nM T64765 CUA2I0 46884425 Ki = 47 nM T64765 CF7HD6 46884426 Ki = 10 nM T64765 C9M4RX 46884427 Ki = 14 nM T64765 CT9K2R 46884428 Ki = 7 nM T64765 C89NXQ 46884429 Ki = 23 nM T64765 CWK75U 46884462 Ki = 7 nM T64765 C82IYB 46884463 Ki = 41 nM T64765 CLX5N1 46884464 Ki = 447 nM T64765 C7K8HU 46884465 Ki > 1000 nM T64765 CU5N4L 46884466 Ki = 560 nM T64765 CGN3O2 46884510 Ki > 1000 nM T64765 CBS8I6 46884511 Ki > 1000 nM T64765 C1X3VT 46884512 Ki > 1000 nM T64765 CZ26BV 46884513 Ki > 1000 nM T64765 C3N9RT 46884514 Ki = 858 nM T64765 CB29TI 46887041 EC50 = 45.71 nM T64765 C9P3CV 46887042 EC50 = 2.884 nM T64765 C12SYH 46887043 EC50 = 5.888 nM T64765 CQJ8W2 46887076 EC50 > 10000 nM T64765 CAG89L 46887077 EC50 > 10000 nM T64765 COK81L 46887078 EC50 > 10000 nM T64765 CB09SD 46887079 EC50 = 4466.84 nM T64765 CK0S2U 46887080 EC50 > 10000 nM T64765 CLPJ52 46887115 EC50 = 2754.23 nM T64765 C7UL8T 46887249 Ki = 8.4 nM T64765 CF4R9M 46887250 Ki = 3.6 nM T64765 CJ0H5B 46887646 Ki = 16 nM T64765 CJ56OW 46887647 Ki = 44 nM T64765 C06VOU 46887700 Ki = 260 nM T64765 C4PQU5 46887701 Ki = 350 nM T64765 C4IG2C 46887702 Ki = 300 nM T64765 CZ1Q0V 46887887 Ki = 5.3 nM T64765 C8IO4F 46887923 Ki = 2.8 nM T64765 C8EOA7 46887961 Ki = 3.4 nM T64765 C0XR8B 46887962 Ki = 1.6 nM T64765 CE4X6C 46887963 Ki = 2 nM T64765 CVB6C0 46887993 Ki = 2.5 nM T64765 C0U3CX 46887994 Ki = 2.4 nM T64765 CG8I9K 46887995 Ki = 3.2 nM T64765 CX7EK0 46887996 Ki = 23 nM T64765 C49VFT 46888006 Ki = 1.1 nM T64765 CMRN14 46888035 Ki = 12 nM T64765 C0UY5G 46888036 Ki = 13 nM T64765 CI1C9M 46888037 Ki = 17 nM T64765 C5E9LR 46888078 Ki = 1.2 nM T64765 CL0TF1 46888079 Ki = 455 nM T64765 CAVC58 46888080 Ki = 51 nM T64765 CFB4L7 46888114 Ki = 16 nM T64765 CC7H5Z 46888115 Ki = 7 nM T64765 C2AWK5 46888161 Ki = 69 nM T64765 CYW38L 46888162 Ki = 150 nM T64765 C29XNB 46888163 Ki = 184 nM T64765 CQ1R2B 46888207 Ki = 50 nM T64765 C48DHL 46888208 Ki = 717 nM T64765 CDN5W1 46888209 Ki = 55 nM T64765 CS3HC4 46888210 Ki = 45 nM T64765 COS18Q 46888267 Ki = 143 nM T64765 C75HYB 46888268 Ki = 89 nM T64765 CDEP03 46888327 Ki = 5.3 nM T64765 CZTO65 46888328 Ki = 4.6 nM T64765 CH7D4U 46888329 Ki = 2.6 nM T64765 CL51ME 46890090 Ki = 7.8 nM T64765 COR71G 46890166 EC50 = 377 nM T64765 C2XCK5 46890181 Ki = 0.6 nM T64765 CTS04G 46890283 Ki = 0.19 nM T64765 CV8C4E 46890347 Ki = 0.05 nM T64765 C4XLV0 46890430 Ki = 0.2 nM T64765 C4IK6F 46890475 Ki = 0.28 nM T64765 CK08VN 46890476 Ki = 0.11 nM T64765 CM56CG 46890523 Ki = 0.22 nM T64765 C2K4HZ 46890562 Ki = 0.69 nM T64765 C89ZNE 46890564 Ki = 12 nM T64765 C8FR9E 46890592 EC50 = 119 nM T64765 CT4Q8R 46890603 Ki = 11 nM T64765 C6XPD3 46890638 Ki = 0.2 nM T64765 CQLS54 46890639 Ki = 3.5 nM T64765 CP7ZS3 46890640 Ki = 0.71 nM T64765 CU3O0K 46890688 Ki = 0.56 nM T64765 C5F1CH 46893542 IC50 = 80 nM T64765 CDV30W 46912441 EC50 = 1.1 nM T64765 CAQ0E9 46912442 Ki = 5.4 nM T64765 CS8HI2 46929441 Ki > 1000 nM T64765 C47HDL 46929447 Ki = 18 nM T64765 CSDO60 46929548 Ki = 530 nM T64765 C06XZG 46929550 EC50 = 48 nM T64765 C6F2MP 46929551 EC50 = 15 nM T64765 CC19QK 46929552 EC50 = 67 nM T64765 CT3UX6 46929553 EC50 = 22 nM T64765 CZJ2G8 46929554 EC50 = 140 nM T64765 C5YC7L 46929556 Ki = 130 nM T64765 C40EGB 46929647 Ki = 14 nM T64765 CB95RA 46929648 EC50 = 74 nM T64765 CQKM36 46930924 Ki > 1000 nM T64765 C9DLV2 46945057 Ki = 5 nM T64765 C71LMB 46945818 Ki = 4.6 nM T64765 CW8YC3 49765184 Ki = 7.4 nM T64765 CQV8C1 49797821 Ki = 11 nM T64765 CFB15T 49797822 Ki = 17 nM T64765 C6Y0FI 49797823 Ki = 41 nM T64765 CCRJ25 49797824 Ki = 5.7 nM T64765 C9OZP7 49799183 Ki = 1.4 nM T64765 CLO87S 49799184 EC50 = 1.6 nM T64765 CAM63P 49799185 Ki = 61 nM T64765 CXPZ46 49799215 Ki = 127 nM T64765 CZMQ60 49799250 Ki > 1000 nM T64765 CO4NP5 49799251 Ki > 1000 nM T64765 CC7TO2 49799253 EC50 = 1.1 nM T64765 C4YT5P 49799254 EC50 = 8.8 nM T64765 C3EWO4 49799506 EC50 = 0.21 nM T64765 C53XBJ 49799507 EC50 = 12 nM T64765 CS53FK 49799508 Ki = 1 nM T64765 C40LMT 49799509 Ki = 14 nM T64765 CJ3Z8H 49799537 Ki = 1.6 nM T64765 CK3MN5 49836075 Ki = 12 nM T64765 CB6OA3 49836197 Ki = 1.6 nM T64765 CP87FO 49836198 Ki = 0.28 nM T64765 CU2NF0 49836199 Ki = 1.4 nM T64765 CFB53A 49836200 Ki = 0.89 nM T64765 CG97QN 49841719 Ki = 188 nM T64765 CZ3T1W 49841845 Ki = 98 nM T64765 C3SBE0 49841846 Ki = 63 nM T64765 CAM2T0 49855508 Ki = 2.8 nM T64765 CQ9X0C 49855509 Ki = 2.1 nM T64765 C61CAO 49855511 Ki = 3.4 nM T64765 C8LBU5 49855513 EC50 = 1 nM T64765 C7LCF8 49855702 Ki = 1170 nM T64765 C4RUN9 49855705 Ki = 19 nM T64765 C79SQV 49855898 Ki > 3000 nM T64765 C16EFA 49855900 Ki = 66 nM T64765 C5F7HI 49856083 Ki = 2 nM T64765 CQ0L4M 49856084 EC50 = 0.9 nM T64765 C42LJP 49856086 Ki = 0.9 nM T64765 CA5DU9 49856277 Ki > 1000 nM T64765 CVR2O7 49856842 Ki = 32 nM T64765 CSZ14T 49857220 Ki = 106 nM T64765 CRO90J 49857807 Ki = 8 nM T64765 C43UWI 49857808 Ki = 10 nM T64765 CC8VZ4 49857811 Ki = 5.4 nM T64765 CPB30Q 49857812 Ki = 100 nM T64765 C0DBR2 49857997 Ki = 6.3 nM T64765 CZO5D6 49857998 EC50 = 1.8 nM T64765 CKO31L 49858001 Ki = 2.5 nM T64765 CM3C2Z 49858196 Ki = 9 nM T64765 C18YTS 49858198 Ki = 9 nM T64765 C8E4MD 49858393 Ki = 3.4 nM T64765 C8QX6M 49859944 Ki = 3.981 nM T64765 CO46BE 49864802 IC50 = 9.2 nM T64765 C8COL5 49864803 IC50 = 3.6 nM T64765 C5BHN9 49864869 IC50 = 5.9 nM T64765 CVH6O7 49864994 IC50 = 20000 nM T64765 CAZ98V 49864995 IC50 = 20000 nM T64765 C4FZD3 49864996 IC50 = 2742 nM T64765 C7GC4R 49864997 IC50 = 25 nM T64765 CZY70R 49865047 IC50 = 738 nM T64765 CLQ1G6 49865048 IC50 = 94 nM T64765 CX49VU 49865109 IC50 = 356 nM T64765 CGUK09 49865110 IC50 = 2.2 nM T64765 C8XF2R 49865111 IC50 = 3.4 nM T64765 CW9DX4 49865112 IC50 = 1761 nM T64765 C7R6EH 49865169 IC50 = 241 nM T64765 C37AYI 49865170 IC50 = 516 nM T64765 C6S9FW 49865171 IC50 = 184 nM T64765 CVX86D 49865172 IC50 = 4894 nM T64765 C7H0ZE 49865226 IC50 = 20000 nM T64765 C3AL7O 49865227 IC50 = 3612 nM T64765 C27TJB 49865228 IC50 = 2431 nM T64765 CG1OE8 49865229 IC50 = 2470 nM T64765 C07RIT 49865289 IC50 = 14215 nM T64765 CR4F9G 49865290 IC50 = 3 nM T64765 CFAE84 49865348 IC50 = 64 nM T64765 CNHI23 49865395 IC50 = 475 nM T64765 C6C7DR 49865396 IC50 = 1891 nM T64765 C5ZP9V 49865448 IC50 = 28 nM T64765 CE8YR7 49865449 IC50 = 14 nM T64765 C1IEH0 49865488 IC50 = 34 nM T64765 C4BF6Q 49865489 IC50 = 19 nM T64765 C35SIM 49865537 IC50 = 0.3 nM T64765 C2RY0J 50878551 Ki = 1698.24 nM T64765 C1W6TV 50898777 Ki > 10000 nM T64765 CXMZ73 50898778 Ki > 10000 nM T64765 CMYP82 50905026 Ki = 3.5 nM T64765 CF0JE8 51003381 Ki = 12 nM T64765 CE4KP1 51050257 Ki > 10000 nM T64765 C1IL7V 51354008 Ki = 380.19 nM T64765 CCX8V5 51354009 Ki = 81.28 nM T64765 CC0QD5 51354010 Ki = 588.84 nM T64765 C2RY8V 51354296 Ki = 380.19 nM T64765 CLFW43 51354297 Ki = 2691.53 nM T64765 CEL4X0 51354298 Ki = 190.55 nM T64765 C3OT2L 51354299 Ki = 104.71 nM T64765 CYHG32 51354300 Ki = 125.89 nM T64765 CDY7Q9 51354301 Ki = 75.86 nM T64765 CQ1S6T 51354302 Ki = 323.59 nM T64765 C1U6YS 51354303 Ki = 70.79 nM T64765 CX8AQ3 51354304 Ki = 36.31 nM T64765 CSHG49 51354581 Ki = 97.72 nM T64765 C8GQM0 51354582 Ki = 60.26 nM T64765 CL0QJ4 51354583 Ki = 112.2 nM T64765 C9S6YJ 51354584 Ki = 91.2 nM T64765 C3UBQ6 51354585 Ki = 114.82 nM T64765 CFG8J0 51354586 Ki = 75.86 nM T64765 C5OC9L 51354587 Ki = 6309.57 nM T64765 C08AOI 51354588 Ki = 18620.87 nM T64765 CI9YD2 51354870 Ki = 794.33 nM T64765 CHN6Q5 51354871 Ki = 489.78 nM T64765 C0V7HN 51354872 Ki = 120.23 nM T64765 CF9V1U 52937018 Ki = 125.89 nM T64765 CS3BJ7 52937119 Ki > 398.11 nM T64765 C93QXP 52937222 Ki = 125.89 nM T64765 CPF7V0 52937223 Ki = 79.43 nM T64765 CYG24L 52937526 Ki = 79.43 nM T64765 CL8QZ3 52937527 Ki = 251.19 nM T64765 CM36PE 52937629 Ki = 316.23 nM T64765 CRV61I 52937630 Ki > 501.19 nM T64765 CEKB47 52937631 Ki > 630.96 nM T64765 CZ0C5B 52937632 Ki > 630.96 nM T64765 CVX7U2 52937633 Ki > 630.96 nM T64765 C3ZX1Q 52937634 Ki > 630.96 nM T64765 CY4N8T 52937728 Ki = 199.53 nM T64765 C83WTP 52937729 Ki > 630.96 nM T64765 CQDS92 52937730 Ki = 630.96 nM T64765 CR0KW9 52937731 Ki = 251.19 nM T64765 C2UV5S 52937732 Ki > 630.96 nM T64765 C6XHP8 52937733 Ki > 630.96 nM T64765 C3B5HN 52937734 Ki = 199.53 nM T64765 CK52QG 52937828 Ki > 1995.26 nM T64765 CFV4D0 52937829 Ki > 630.96 nM T64765 C9MBQ2 52937830 Ki > 398.11 nM T64765 C19EOL 52941001 Ki = 520 nM T64765 CFL5N7 52941024 IC50 = 2 nM T64765 CG63NI 52941057 IC50 = 9 nM T64765 CE9F1Q 52941061 IC50 = 41 nM T64765 C29BFI 52941062 IC50 = 5508 nM T64765 CQW15U 52941269 Ki = 9 nM T64765 C6FTJ8 52941311 Ki = 14 nM T64765 C63HFA 52941318 Ki = 24 nM T64765 CM9D2S 52941450 Ki > 1000 nM T64765 C73SKO 52941508 Ki > 3000 nM T64765 CB9RQ8 52941660 Ki = 0.9 nM T64765 C6AG2P 52941662 Ki = 261 nM T64765 CTZ65F 52942159 Ki > 1000 nM T64765 CL36BN 52942843 IC50 = 2 nM T64765 CL9QT8 52942844 Ki = 3280 nM T64765 CTN09Z 52943330 IC50 = 709 nM T64765 C4BLG0 52943401 Ki = 2130 nM T64765 CH87IQ 52943448 IC50 = 17 nM T64765 CWY91T 52943449 IC50 = 84 nM T64765 CH42FY 52943741 Ki = 155 nM T64765 C14EYP 52943742 Ki > 1000 nM T64765 CH6A8X 52943846 Ki = 93 nM T64765 CPR7I5 52943847 Ki = 41 nM T64765 CY0VU3 52944348 Ki = 187 nM T64765 CUL0T9 52944521 IC50 = 12 nM T64765 CTI28E 52944579 Ki = 4 nM T64765 CKI59T 52944686 IC50 = 20 nM T64765 C6PNI0 52945858 IC50 = 14 nM T64765 CEFC04 52946273 Ki = 110 nM T64765 CM30FQ 52946282 Ki = 7.4 nM T64765 C9OC6P 52946526 Ki = 50 nM T64765 CX70CR 52947031 Ki = 257 nM T64765 CWRV27 52947715 Ki = 153 nM T64765 CCN9H6 52947729 Ki > 1000 nM T64765 CG3QP5 52948008 Ki = 17 nM T64765 C48JMX 52948255 Ki = 2 nM T64765 CB1CM6 52948312 Ki = 15 nM T64765 CN16EQ 52948626 Ki = 344 nM T64765 C3VR4X 52948730 Ki = 32 nM T64765 C1G9CV 52949835 Ki = 357 nM T64765 C2HC4G 52949865 Ki = 20 nM T64765 CC2Q0P 52952957 Ki = 239.88 nM T64765 CVT41A 53317856 Ki = 48.6 nM T64765 CGT13D 53317857 Ki = 60 nM T64765 C7UY4X 53317858 Ki = 30 nM T64765 CND27K 53317859 Ki = 40.1 nM T64765 CI7C5Y 53318961 Ki = 31.9 nM T64765 CB8L6U 53319170 Ki = 4 nM T64765 C73ZRL 53319171 Ki = 163 nM T64765 C7HC3A 53320008 Ki = 65 nM T64765 CC7KB2 53320488 Ki = 42.6 nM T64765 CKPN38 53320489 Ki = 15 nM T64765 C07QLD 53320490 Ki = 652.6 nM T64765 C61MCX 53320491 Ki = 36 nM T64765 C3Z4LB 53321787 Ki = 80.1 nM T64765 C2M3KN 53321788 Ki = 23 nM T64765 CQ67PM 53321789 Ki = 36 nM T64765 C1S3BX 53321790 Ki = 39 nM T64765 CPYV96 53321791 Ki = 161 nM T64765 C1L7WJ 53321919 EC50 = 0.3981 nM T64765 CDN71E 53323110 Ki = 12 nM T64765 CQ5N8A 53323111 Ki = 50 nM T64765 CC7LW8 53323112 Ki = 40 nM T64765 CI3MX0 53324463 Ki = 49 nM T64765 C2JLF0 53324464 Ki = 6.1 nM T64765 CXHS51 53324465 Ki = 28 nM T64765 CIK14U 53324466 Ki = 161.8 nM T64765 C78TYH 53325775 Ki = 62 nM T64765 CX63DZ 53325776 Ki = 72 nM T64765 CQ04OC 53325777 Ki = 16 nM T64765 C1UT3Q 53325778 Ki = 182.3 nM T64765 CD8IP1 53325779 Ki = 36.4 nM T64765 CBG60V 53326914 Ki = 69 nM T64765 CU59EZ 53363442 EC50 = 1.1 nM T64765 C5C3TQ 53363444 Ki = 82 nM T64765 CQA21I 53363445 Ki = 16 nM T64765 CME4F1 53363446 Ki = 16 nM T64765 CN5JP2 53363447 Ki = 767 nM T64765 C1YEN6 53363717 Ki = 3.9 nM T64765 CV16AX 53363718 Ki = 4.8 nM T64765 CXC7N1 53363719 Ki = 2.5 nM T64765 CB3DN2 53363720 Ki = 6.9 nM T64765 C06SOJ 53363721 Ki = 21 nM T64765 C52LEA 53363722 Ki = 9.2 nM T64765 CX5L8D 53363808 Ki = 295 nM T64765 CMOZ61 53475319 Ki = 893 nM T64765 CFU8T7 53483937 EC50 = 1.3 nM T64765 CZBK68 53530230 IC50 = 2190 nM T64765 CYM2T4 53868701 Ki = 87 nM T64765 CZ34PR 54584374 Ki = 549.54 nM T64765 CFDA28 54584378 Ki = 257.04 nM T64765 CYF4K3 54587323 Ki = 26 nM T64765 CELM42 54587325 Ki = 20 nM T64765 CD8YN4 54753626 Ki = 0.4 nM T64765 CL32AY 54753627 Ki = 0.5 nM T64765 CB72FX 54754351 Ki = 646 nM T64765 CPS5V6 54764158 Ki = 0.7 nM T64765 C9OUQ6 54765288 IC50 = 189.3 nM T64765 CZJ3B1 56648033 Ki = 3.3 nM T64765 CP2B8C 56657939 Ki = 3.6 nM T64765 CHX56Z 56658414 Ki = 15 nM T64765 CG2OI0 56658415 Ki = 210 nM T64765 CTKN69 56658545 Ki = 1120 nM T64765 CPJ7D3 56658546 Ki = 2.3 nM T64765 C7AG6I 56658547 Ki = 0.8 nM T64765 C6W5UT 56658548 Ki = 1.5 nM T64765 CFTE47 56658571 Ki > 10000 nM T64765 C71XNV 56658572 Ki = 3.5 nM T64765 CP1OV6 56658588 Ki = 0.32 nM T64765 C9TFO2 56658589 Ki = 0.53 nM T64765 CL2YE8 56659224 Ki = 1.6 nM T64765 C5F1TD 56659225 Ki = 1.5 nM T64765 CFD6N4 56659892 Ki = 10 nM T64765 CZSM65 56659893 Ki = 16 nM T64765 CM6A3K 56661468 Ki = 1.8 nM T64765 C8ZRL1 56661905 Ki > 1000 nM T64765 CKUI61 56661999 Ki = 11 nM T64765 C2QTH5 56662000 Ki = 2.6 nM T64765 CTOP89 56662001 Ki = 23 nM T64765 C9F5WK 56662040 Ki = 0.25 nM T64765 CCEO61 56662041 Ki = 0.64 nM T64765 CO3I1H 56662705 Ki = 3.4 nM T64765 CJ9RG0 56663350 Ki = 3.4 nM T64765 C1GZM7 56663405 Ki = 2.4 nM T64765 C3XW6G 56664901 Ki = 1.6 nM T64765 C9WDB6 56664902 Ki = 0.3 nM T64765 CC1GK4 56665357 Ki = 0.8 nM T64765 C7W1LB 56665358 Ki = 1.4 nM T64765 C7A0UB 56665493 Ki = 48 nM T64765 CMY64U 56665506 Ki = 4.2 nM T64765 C7CG0S 56665507 Ki = 21 nM T64765 CM07UW 56665518 Ki = 5.5 nM T64765 CL4XG3 56666171 Ki = 2.5 nM T64765 CHB63V 56666239 Ki = 1 nM T64765 CMZ6K8 56666240 Ki = 5 nM T64765 CT37LU 56668326 Ki = 2.8 nM T64765 CJ95CA 56668427 Ki = 1.4 nM T64765 CQR32B 56668530 Ki = 5.2 nM T64765 C3L7FD 56668789 Ki = 0.8 nM T64765 C7MR5P 56668790 Ki = 1.7 nM T64765 CJ37DR 56668799 Ki = 173 nM T64765 C3YVL9 56668800 Ki = 184 nM T64765 CH0V1I 56668921 Ki = 50 nM T64765 CS79GB 56668922 Ki = 1.5 nM T64765 CM03XH 56668952 Ki = 0.56 nM T64765 C25HCW 56668953 Ki = 0.26 nM T64765 C4NR8W 56669644 Ki = 3.5 nM T64765 C5K4NS 56670257 Ki = 37 nM T64765 C8XSR7 56670466 Ki = 38 nM T64765 CY0GX2 56671810 Ki = 3.6 nM T64765 C2GFT1 56671811 Ki = 1.6 nM T64765 CCI1K3 56671812 Ki = 8.3 nM T64765 C6LQ1R 56672280 Ki = 15 nM T64765 CQ0JD6 56672398 Ki = 23 nM T64765 CD91TO 56672437 Ki = 3.2 nM T64765 CP9Z2L 56673090 Ki = 2 nM T64765 C83MQK 56673091 Ki = 4 nM T64765 CC04NV 56673156 Ki = 0.7 nM T64765 C6FPR7 56673157 Ki = 2.5 nM T64765 C5G0ID 56673158 Ki = 1 nM T64765 CX7RI0 56675667 Ki = 4 nM T64765 C8OEI6 56675668 Ki = 7 nM T64765 C6ANT4 56675784 Ki = 4.6 nM T64765 CC9Y6F 56675822 Ki = 0.57 nM T64765 C4B5JQ 56675823 Ki = 0.17 nM T64765 CP41OM 56676397 Ki = 1.6 nM T64765 CWS95P 56676398 Ki = 6.31 nM T64765 CSRV63 56677109 Ki = 110 nM T64765 CZP86D 56677285 EC50 = 2.1 nM T64765 C5M0AS 56678518 Ki = 4.8 nM T64765 C7IWP6 56678519 Ki = 2.5 nM T64765 C0IGC6 56678520 Ki = 4.9 nM T64765 CT7BE0 56678521 Ki = 2.2 nM T64765 C8QOB7 56678653 Ki = 5 nM T64765 CY5HJ2 56678654 Ki = 9 nM T64765 CN9IV8 56678977 Ki = 9 nM T64765 C40NBA 56679098 Ki = 1.9 nM T64765 C46ZSY 56679099 Ki = 4 nM T64765 CRF3V7 56679100 Ki = 2.4 nM T64765 CW7QF9 56679101 Ki = 1.6 nM T64765 C0NAF1 56679117 Ki = 15 nM T64765 CO4V1S 56679118 Ki = 49 nM T64765 CSHO51 56679737 Ki = 2.4 nM T64765 C6DHC5 56680370 Ki = 5.7 nM T64765 C0O8YP 56680371 Ki = 152 nM T64765 CZ2AM6 56680431 Ki > 500 nM T64765 C4MH8J 56681858 Ki = 5.2 nM T64765 CC4N7R 56682288 Ki = 84 nM T64765 CT3OI2 56682300 Ki = 3.6 nM T64765 C7F1JG 56683065 Ki = 1.6 nM T64765 CJC19B 56683709 Ki = 2.9 nM T64765 CIY31D 56683751 Ki = 3 nM T64765 C2BE0Y 56683753 Ki = 93 nM T64765 C07ZGE 56683754 Ki = 308 nM T64765 CY92VU 56835087 Ki = 4 nM T64765 C0JMA7 56835088 Ki = 7 nM T64765 CR7LS4 56835090 EC50 = 0.73 nM T64765 C4E6HV 56835171 Ki = 3388.44 nM T64765 CND5M6 56849569 Ki = 1.622 nM T64765 C6Y4GM 56849571 Ki = 1.148 nM T64765 C7YVT9 56851441 Ki = 42.66 nM T64765 CN0P6H 56851443 Ki = 9.772 nM T64765 C7VE0O 56851445 Ki = 46.77 nM T64765 CBW34E 56851447 Ki = 1.023 nM T64765 C6XG8Z 56851602 Ki = 4.898 nM T64765 CQ51VT 56851604 Ki = 16.98 nM T64765 CGO4X5 56851606 Ki = 32.36 nM T64765 C4QHS9 56851608 Ki = 18.62 nM T64765 CQOE56 56851610 Ki = 67.61 nM T64765 CCO25Y 56851612 Ki = 4.677 nM T64765 C7B8RI 56954318 EC50 > 10000 nM T64765 C7G3TI 56954320 EC50 = 4.169 nM T64765 CKG35O 56954322 EC50 = 1.778 nM T64765 CI7XO6 56954425 EC50 > 1000 nM T64765 C2W9CZ 56954427 EC50 = 446.68 nM T64765 CIQH95 56954515 EC50 = 2.884 nM T64765 C1TC7Q 56963799 Ki = 0.4 nM T64765 CDB1F6 57327814 Ki = 4 nM T64765 CO9RV4 57328003 Ki = 1.479 nM T64765 CS2PJ1 57328076 Ki = 0.6607 nM T64765 CYHP54 57328077 Ki = 19.05 nM T64765 C9TOC0 57328078 Ki = 16.6 nM T64765 CW1YS8 57328079 Ki = 5.623 nM T64765 C5J8EQ 57328080 Ki = 1.288 nM T64765 C4HUF2 57328081 Ki = 2.344 nM T64765 C50CFD 57328141 Ki = 2.455 nM T64765 CKB8T1 57328142 Ki = 1.549 nM T64765 CT92DL 57328143 Ki = 1.259 nM T64765 CEO74T 57328144 Ki = 3.02 nM T64765 CD5GS3 57328145 Ki = 2.455 nM T64765 C25AFJ 57328146 Ki = 1.995 nM T64765 CG80ZN 57328209 Ki = 0.871 nM T64765 CT2F3I 57328210 Ki = 0.5129 nM T64765 C2DF8K 57328211 Ki = 2.57 nM T64765 C0QDE3 57328212 Ki = 1.259 nM T64765 CS25HQ 57328213 Ki = 2.042 nM T64765 CR1L2W 57328276 Ki = 12882.5 nM T64765 CFE9O8 57328277 Ki = 13489.63 nM T64765 CT8VZ6 57345658 Ki = 7 nM T64765 C7O0AI 57345659 Ki = 9 nM T64765 C3L9ZA 57345660 Ki = 2 nM T64765 CZK3M1 57345661 Ki = 6 nM T64765 CV89XN 57384004 Ki = 3 nM T64765 C1QDY5 57390430 Ki = 260 nM T64765 CWP8G7 57390431 Ki = 37 nM T64765 CXWZ39 57390432 Ki = 23 nM T64765 CPH4D6 57390433 Ki = 119 nM T64765 C9KL7U 57390469 Ki = 79 nM T64765 C9ZY5S 57390580 Ki = 4.9 nM T64765 CJ7F1T 57390581 Ki = 1.8 nM T64765 C32MYT 57390798 Ki = 4.4 nM T64765 CUHD62 57390842 Ki = 695 nM T64765 C06AFO 57391841 Ki = 18 nM T64765 CGR5M2 57391842 Ki = 12 nM T64765 CEK3U0 57392213 Ki = 150 nM T64765 CJL2R5 57392214 Ki = 278 nM T64765 C5MQ1J 57392215 Ki = 70 nM T64765 CD7C4V 57392216 Ki = 43 nM T64765 CSYC20 57392253 Ki = 117 nM T64765 C6C1WO 57392357 Ki = 37 nM T64765 CO1V0I 57392412 IC50 = 52.4 nM T64765 C4J9FZ 57392413 IC50 = 182 nM T64765 CAL75E 57392460 Ki = 36600 nM T64765 C46NRA 57392651 Ki = 4 nM T64765 C3YV7C 57392890 Ki = 2500 nM T64765 CD5R1S 57393207 Ki = 0.9 nM T64765 CDM8Z6 57393208 Ki = 112 nM T64765 CJ70FG 57393505 Ki = 15 nM T64765 CEQ61P 57393572 Ki = 23 nM T64765 CMSO52 57393969 Ki = 1526 nM T64765 C0WD9F 57393970 Ki = 37 nM T64765 CR72CB 57394133 IC50 = 129.7 nM T64765 CZSU79 57394626 Ki = 13600 nM T64765 C7CWP2 57394928 Ki = 3.5 nM T64765 CF4A6M 57395538 Ki = 17900 nM T64765 CI5M2U 57395620 Ki = 8220 nM T64765 C8F0QY 57395712 Ki = 233 nM T64765 CV18DS 57395713 Ki = 249 nM T64765 C5NY9S 57395714 Ki = 238 nM T64765 CBAU35 57395715 Ki = 58 nM T64765 CAF8N9 57395716 Ki = 25 nM T64765 CNLP18 57395717 Ki = 18 nM T64765 C6Y1RI 57395870 Ki = 38 nM T64765 CT9Z5R 57395871 Ki = 2 nM T64765 CFE50K 57395872 Ki = 21 nM T64765 CY6BP7 57395916 IC50 = 170.6 nM T64765 C38AIS 57396087 EC50 = 1.3 nM T64765 CTI36W 57396117 Ki = 6 nM T64765 CVC80A 57396684 Ki = 3.4 nM T64765 C8ZSN5 57397054 Ki = 23 nM T64765 CXT3G1 57397506 Ki = 379 nM T64765 C6JSX7 57397508 Ki = 357 nM T64765 CIR5B4 57397509 Ki = 95 nM T64765 C4PXI8 57397510 Ki = 47 nM T64765 C87BYX 57397650 Ki = 7.7 nM T64765 CQS0M5 57397654 EC50 = 1.3 nM T64765 C9Y6KG 57397934 Ki = 4 nM T64765 CRDW25 57398452 Ki = 2 nM T64765 CA4ET0 57398826 Ki = 42 nM T64765 CS18MF 57398827 Ki = 15 nM T64765 CLOZ63 57399127 Ki = 196 nM T64765 C9I8JL 57399192 Ki = 15 nM T64765 CRW37S 57399193 Ki = 79 nM T64765 CH80GZ 57399194 Ki = 33 nM T64765 C4ZV7N 57399234 Ki = 109 nM T64765 CCSL05 57399326 Ki = 9 nM T64765 COUZ23 57399327 Ki = 5 nM T64765 CO5H6E 57399328 Ki = 10 nM T64765 CHJ64B 57399329 Ki = 20 nM T64765 C6ORJ9 57399371 IC50 = 260 nM T64765 CBZ51V 57400497 Ki = 38 nM T64765 C6HS9E 57400498 Ki = 39 nM T64765 CV53MQ 57400499 Ki = 17 nM T64765 CZ7AG2 57400500 Ki = 18 nM T64765 CP75KQ 57400777 Ki = 8750 nM T64765 C06WSZ 57400778 Ki = 15500 nM T64765 C07SNI 57400950 Ki = 288 nM T64765 CCF54S 57400951 Ki = 15 nM T64765 CX17EI 57400952 Ki = 35 nM T64765 CI7CK1 57401087 Ki = 18 nM T64765 C4TOX0 57401094 Ki = 5 nM T64765 C0VXJ4 57401342 Ki = 9.2 nM T64765 CD8BA0 57402310 Ki = 126 nM T64765 CR6WS7 57402311 Ki = 25 nM T64765 C9DOI4 57402312 Ki = 27 nM T64765 C1BLC9 57402706 Ki = 370 nM T64765 CKA35J 57402707 Ki = 36 nM T64765 CJ8IW2 57402708 Ki = 143 nM T64765 C2CFA9 57402849 Ki = 74 nM T64765 CVLW85 57402850 Ki = 8.8 nM T64765 C10PXB 57402928 Ki = 28600 nM T64765 C65TPY 57403054 EC50 = 1.6 nM T64765 C1JFL4 57403350 Ki = 825 nM T64765 CM2UK4 57403351 Ki = 54 nM T64765 CNEI24 57403650 Ki = 4.7 nM T64765 CLH73S 57404025 Ki = 15 nM T64765 CF5R2M 57404026 Ki = 26 nM T64765 C4RHF3 57404027 Ki = 10 nM T64765 CT94RI 57404028 Ki = 15 nM T64765 CRL2O8 57404029 Ki = 16 nM T64765 CUOV05 57411066 Ki = 3 nM T64765 C7AMZ8 57437617 Ki > 10000 nM T64765 CO4ZY2 57612982 Ki = 7.8 nM T64765 C9R0MA 57672010 Ki = 19 nM T64765 C0UAD2 57672016 Ki = 0.23 nM T64765 CE3G4X 57672043 Ki = 0.17 nM T64765 CF3IK6 57755473 Ki = 0.5012 nM T64765 CT89JH 57780007 Ki = 1.995 nM T64765 CT8RO7 57780008 Ki = 0.5012 nM T64765 C5RIN4 57780016 Ki = 1.585 nM T64765 CE9WC0 57780017 Ki = 1.585 nM T64765 C1W4SB 57780018 Ki = 1.259 nM T64765 CT96WD 57780020 Ki = 0.7943 nM T64765 CXI6A1 57970302 IC50 = 930 nM T64765 CSTV53 58198951 Ki = 7 nM T64765 CPY01C 58198985 Ki = 3 nM T64765 CBZX94 58199027 Ki = 4 nM T64765 CL6B2G 58199044 Ki = 47 nM T64765 C2E8AM 58199450 Ki = 7 nM T64765 CH50YQ 58285100 Ki = 7 nM T64765 CUX9D6 58430446 Ki = 22.8 nM T64765 CIE6Z2 58430454 Ki = 53 nM T64765 CX7V8T 58430485 Ki = 82.8 nM T64765 CLQT57 58430524 Ki = 61 nM T64765 CUTR41 58430577 Ki = 20 nM T64765 CPZH02 58430604 Ki = 13 nM T64765 C7VDB1 58430625 Ki = 15 nM T64765 CXD71J 58430683 Ki = 10 nM T64765 C19QNY 58430684 Ki = 17.8 nM T64765 CE5ZI7 58430715 Ki = 192.4 nM T64765 C4MTV8 58430749 Ki = 12.7 nM T64765 CB3NP1 58430778 Ki = 16.5 nM T64765 CUY96F 58430796 Ki = 78.9 nM T64765 C3AC4U 58430801 Ki = 35.9 nM T64765 CF1OW7 58430814 Ki = 34 nM T64765 CNUT13 59218182 Ki = 1.3 nM T64765 CHVU94 59218184 Ki = 1.5 nM T64765 CY6EB4 59218190 Ki = 0.7 nM T64765 CK4Y8T 59395224 IC50 = 360 nM T64765 CFDG19 59401765 IC50 = 0.71 nM T64765 CF65GP 59401771 IC50 = 0.48 nM T64765 CC5QW1 59401793 IC50 = 0.66 nM T64765 CQK9S3 59401826 Ki = 13.8 nM T64765 C53BVH 59401876 Ki = 8.6 nM T64765 CNOI48 59401886 IC50 = 0.0092 nM T64765 CA9NE4 59548712 Ki = 2.3 nM T64765 C78LMC 59548713 Ki = 3.5 nM T64765 CAD1J6 59589020 Ki > 3000 nM T64765 CAM03U 59651897 Ki = 5 nM T64765 CT36HR 59651902 Ki = 16 nM T64765 CS5K7T 59651911 Ki = 25 nM T64765 CYKF93 59651916 Ki = 4 nM T64765 C6SW0N 59651954 Ki = 4.7 nM T64765 C5PDB3 59651957 EC50 = 1.7 nM T64765 CE5O2G 59651983 Ki = 20 nM T64765 C5UPD1 59651984 Ki = 4 nM T64765 C4W8RH 59651989 Ki = 3.7 nM T64765 C04REG 59651991 Ki = 3.7 nM T64765 CP5UN4 59651998 Ki = 47 nM T64765 CIL17E 59652016 Ki = 17 nM T64765 C5T7JX 59652019 Ki = 10 nM T64765 CW5LS2 59652024 Ki = 4.3 nM T64765 CW59BZ 59652026 Ki = 6.9 nM T64765 C0BN4G 59652033 Ki = 3.6 nM T64765 CDP47R 59652049 Ki = 105 nM T64765 C8JZP7 59652054 Ki = 15 nM T64765 C08TLU 59652056 Ki = 27 nM T64765 CV3F5G 59652059 Ki = 4.5 nM T64765 CI74MC 59777245 EC50 = 79.43 nM T64765 CNKF60 60143411 IC50 = 10000 nM T64765 CYCN68 60143412 IC50 = 6060 nM T64765 CJP6A3 60143413 IC50 = 8310 nM T64765 CX9PB5 60143414 IC50 = 16500 nM T64765 CGJ5H3 60143415 IC50 = 1330 nM T64765 C7TC5K 60143416 IC50 = 830 nM T64765 CRFV62 60143588 IC50 = 2570 nM T64765 C7S4PH 60143589 IC50 = 1740 nM T64765 C9EH3R 60143590 IC50 = 91100 nM T64765 CZ3QD9 60143591 IC50 = 19600 nM T64765 CM62NL 60143592 IC50 = 18000 nM T64765 C9ME8V 60143757 IC50 = 29900 nM T64765 CFH4L9 60143758 IC50 = 17500 nM T64765 C4R6PH 60143759 IC50 = 22600 nM T64765 CVA2X8 60143760 IC50 = 18500 nM T64765 CD65CK 60143761 IC50 = 4850 nM T64765 C4TES3 60143762 IC50 > 10000000 nM T64765 CR1ZN4 60143921 IC50 = 13200 nM T64765 CD5T7O 60143922 IC50 = 10000 nM T64765 C5DJA6 60143923 IC50 > 100000000 nM T64765 CPF6A9 60143924 IC50 = 11800 nM T64765 CRTN28 60143925 IC50 = 400 nM T64765 CYJ19Q 60143926 IC50 = 320 nM T64765 C8UQ7D 60144084 IC50 = 500 nM T64765 CPLG49 60144085 IC50 = 500 nM T64765 CM0C9O 60144086 IC50 = 10400 nM T64765 C03VOZ 60144087 IC50 = 20900 nM T64765 CN4A8W 60144088 IC50 = 29800 nM T64765 CJ4XM3 60144089 IC50 = 320 nM T64765 CY4H9Z 60144244 IC50 = 400 nM T64765 CMQ78O 60144245 IC50 = 500 nM T64765 C4NZ3G 60145489 IC50 = 250 nM T64765 CAPO85 60145490 IC50 > 10000000 nM T64765 C8W0YT 60145491 IC50 = 400 nM T64765 C4KZ3M 60145492 IC50 = 700 nM T64765 CBP2K4 60145493 IC50 = 390 nM T64765 C0B7QX 60145494 IC50 > 10000000 nM T64765 CDK1O7 60145629 IC50 > 100000000 nM T64765 COR56Z 60145630 IC50 = 88600 nM T64765 C03HNY 60145631 IC50 > 10000000 nM T64765 C6CE5G 60145632 IC50 > 10000000 nM T64765 CJSV45 60145633 IC50 = 107000 nM T64765 CB4ND5 60145634 IC50 = 16600 nM T64765 C0FR9I 60145771 IC50 = 53800 nM T64765 C8S4EL 60145772 IC50 = 93600 nM T64765 CE17ZH 60145773 IC50 = 82000 nM T64765 CHJ03O 60145774 IC50 = 77900 nM T64765 C40GSO 60145775 IC50 = 13400 nM T64765 CG6F4M 60145776 IC50 = 164 nM T64765 CSNZ26 60150162 Ki = 158.49 nM T64765 C9YP3F 60150166 Ki = 144.54 nM T64765 CTL97W 60151476 Ki = 8.73 nM T64765 C90BYF 60196780 Ki = 14.9 nM T64765 CGBT45 60196783 Ki = 4.1 nM T64765 CF0TM3 60196786 Ki = 3.8 nM T64765 C3YKM9 60196875 Ki = 26.9 nM T64765 CT7CK8 60196882 Ki = 5.39 nM T64765 CEO6K0 60196884 Ki = 62.04 nM T64765 C1TMK4 60196979 Ki = 14.8 nM T64765 CWG0V5 60196980 Ki = 29.91 nM T64765 CIO5W3 60196981 Ki = 75.8 nM T64765 C03SMV 60197083 Ki = 4.89 nM T64765 CI05HA 60197085 Ki = 2.4 nM T64765 CHR18U 60197086 Ki = 90.75 nM T64765 CT2N3E 60197280 Ki = 4.05 nM T64765 CPKR45 62705087 Ki = 66 nM T64765 CLIN39 62705088 Ki = 12 nM T64765 CWMD31 62705089 Ki = 14 nM T64765 C2Q4BR 62705090 Ki = 3 nM T64765 C7VYR4 62705091 Ki = 11 nM T64765 C0PRJ4 62705249 Ki = 53 nM T64765 CD4OF0 62705250 Ki = 4 nM T64765 C7ZST6 62705251 Ki = 67 nM T64765 CMBX94 62705252 Ki = 8 nM T64765 CO9I0P 62707524 Ki = 30 nM T64765 CV76SE 62707525 Ki = 120 nM T64765 C7WZA4 62707526 Ki = 37 nM T64765 C8C2UP 62707527 Ki = 46 nM T64765 C4R8OG 67401728 IC50 = 0.006 nM T64765 CNS9A4 68227454 Ki = 4.2 nM T64765 C95KFZ 68269754 Ki = 0.6 nM T64765 C68RYQ 68269759 Ki = 4 nM T64765 CCL07A 68269762 Ki = 1.2 nM T64765 CT65CN 68269765 Ki = 3.9 nM T64765 CG57KV 68269767 Ki = 4.6 nM T64765 CP74ZW 68269773 Ki = 3 nM T64765 CI6YC4 68378925 IC50 > 30000 nM T64765 CI7S6T 68378958 IC50 > 30000 nM T64765 CU71NC 68379030 IC50 > 30000 nM T64765 C7CBD4 68379135 IC50 > 30000 nM T64765 CT32VB 68379165 IC50 > 30000 nM T64765 CBD8C9 68379213 IC50 = 860 nM T64765 CY35OF 68497905 Ki = 2.5 nM T64765 CR8S1L 68504529 Ki = 1.259 nM T64765 CLA87B 68504537 Ki = 0.5012 nM T64765 C36YVI 68504544 Ki = 0.1259 nM T64765 CLFT03 68504950 Ki = 0.5012 nM T64765 CD4T2F 68506105 Ki = 0.3162 nM T64765 CJ2F6B 68506266 Ki = 1.585 nM T64765 C7EX0S 68506719 Ki = 0.1995 nM T64765 C1XNP4 68506820 Ki = 0.631 nM T64765 C58QHP 68507598 Ki = 0.631 nM T64765 C4Y8GH 68507915 Ki = 1.585 nM T64765 C7P9WX 68508016 Ki = 2.512 nM T64765 C47AGJ 68509493 Ki = 2.512 nM T64765 C20LBF 68509511 Ki = 0.5012 nM T64765 C4DN7V 68511788 Ki = 0.7943 nM T64765 C1XL6P 68511915 Ki = 0.3981 nM T64765 CYV20U 68728631 Ki = 1.7 nM T64765 CD3U6K 68731121 Ki = 1.7 nM T64765 C6IP8Q 69082816 Ki = 1.7 nM T64765 C51SBU 69094686 Ki = 0.2512 nM T64765 C69ZCT 69189076 Ki = 6.9 nM T64765 CSO13P 69248099 Ki = 316.23 nM T64765 CH3SB0 69355600 Ki = 4.074 nM T64765 C7R2WX 69744095 Ki = 159 nM T64765 C2IN4A 70681643 Ki = 23.8 nM T64765 C8HF3M 70685675 IC50 = 130 nM T64765 C91SZE 70685900 Ki = 3.4 nM T64765 COZN69 70687957 Ki = 7769 nM T64765 CG3AL0 70688023 Ki = 4.4 nM T64765 C4G7IY 70690039 Ki = 4.2 nM T64765 CJX1W4 70694267 Ki = 24.5 nM T64765 CGD95I 70694268 Ki = 3.2 nM T64765 CWZ9I4 70696358 Ki = 29 nM T64765 CD0S8J 71272312 Ki = 230 nM T64765 CM6G3W 71272563 Ki = 1371 nM T64765 C2DR0G 71276378 Ki = 21 nM T64765 CBWP45 71276381 Ki = 530 nM T64765 C0GL4U 71276387 Ki = 9 nM T64765 CV7ZP5 71276437 Ki = 9 nM T64765 C8OGT4 71283628 IC50 = 5000 nM T64765 CBQ8P4 71449250 Ki = 398.11 nM T64765 CE6YD5 71450707 Ki = 5500 nM T64765 CDI84E 71450922 IC50 > 10000 nM T64765 CB83YL 71451044 Ki = 630.96 nM T64765 C0YXD3 71452871 Ki = 630.96 nM T64765 CY7NM9 71452872 Ki = 251.19 nM T64765 C4X9KY 71454294 Ki > 10000 nM T64765 CA65OQ 71454295 Ki > 10000 nM T64765 C4JN5I 71454639 Ki = 630.96 nM T64765 CFBC49 71455896 Ki > 10000 nM T64765 CD4HQ6 71456045 Ki > 10000 nM T64765 CD78KL 71456046 Ki > 10000 nM T64765 CMBU21 71456359 Ki = 398.11 nM T64765 CVT39B 71456360 Ki = 630.96 nM T64765 CK87DI 71456361 Ki = 630.96 nM T64765 CSX5J0 71457844 Ki > 10000 nM T64765 C3VMS0 71458203 Ki = 398.11 nM T64765 C8T5EJ 71458204 Ki = 316.23 nM T64765 CZ6BX7 71458205 Ki = 630.96 nM T64765 CD10CQ 71459761 Ki > 10000 nM T64765 CWM41R 71459943 Ki = 2.884 nM T64765 CDYJ07 71461659 Ki = 5.495 nM T64765 C2OD4S 71461660 Ki = 3.89 nM T64765 CEBC62 71461781 Ki = 436.52 nM T64765 C9DJ1V 71461782 Ki = 630.96 nM T64765 CM7VD9 71519012 Ki = 84660 nM T64765 CLQ31I 71519674 Ki = 630.96 nM T64765 C8JC6A 71525586 Ki = 213.8 nM T64765 CR9ZE5 71525587 Ki = 9549.93 nM T64765 CRL42M 71525588 Ki = 831.76 nM T64765 CZ0FT2 71525589 Ki = 144.54 nM T64765 CRM9Q1 71525678 Ki = 776.25 nM T64765 C2GK7O 71525679 Ki = 1513.56 nM T64765 C7HR1A 71525680 Ki = 1000 nM T64765 C8A0NC 71525681 Ki = 151.36 nM T64765 CE92DF 71528209 Ki = 6.51 nM T64765 C3O6EK 71529541 Ki = 3 nM T64765 C74DBP 71529576 Ki = 43 nM T64765 CO2K1J 71601549 Ki = 6.8 nM T64765 C3W6IK 71601550 Ki = 8.6 nM T64765 C54YIV 71601692 Ki = 1.4 nM T64765 CVU51E 71601693 Ki = 18 nM T64765 C35FSE 71601694 Ki = 3.9 nM T64765 COW2Z6 71601695 Ki = 4.1 nM T64765 C2NE5K 71601696 Ki = 2.9 nM T64765 C8ER2U 71601697 Ki = 13 nM T64765 C3VH1S 71601698 Ki = 3.3 nM T64765 CWY6V7 71601842 Ki = 4 nM T64765 CZ1W3A 71601843 Ki = 15 nM T64765 C84JWF 71601844 Ki = 1.9 nM T64765 C3XKL2 71603135 Ki = 331.13 nM T64765 CQ3Y9W 71603136 Ki = 158.49 nM T64765 CT8WF0 71603137 Ki = 851.14 nM T64765 CDW08C 71603138 Ki = 489.78 nM T64765 CA4GQ7 71603139 Ki = 154.88 nM T64765 CK4T5Q 71603140 Ki = 691.83 nM T64765 C70OBY 71603141 Ki = 218.78 nM T64765 C1HEY4 71603142 Ki = 616.6 nM T64765 CUW27Q 71603194 Ki = 602.56 nM T64765 CO2P7E 71603195 Ki = 177.83 nM T64765 CE0SI2 71625480 IC50 = 73.1 nM T64765 C1N0UT 71625481 IC50 = 14.7 nM T64765 CIL40N 71625482 IC50 = 16.4 nM T64765 CLK47W 71625594 IC50 = 39.1 nM T64765 C4SG8H 71625595 IC50 = 148.6 nM T64765 C1LYR0 71625596 IC50 = 111.4 nM T64765 C2Q1RW 71625597 IC50 = 7.9 nM T64765 C18AQF 71625598 IC50 = 9.1 nM T64765 C4Q9GD 71625599 IC50 = 1 nM T64765 CQC03U 71625710 IC50 = 0.7 nM T64765 C0YW3T 71625711 IC50 = 0.5 nM T64765 CE6DB2 71625712 IC50 = 0.2 nM T64765 CLR3A0 71625825 IC50 = 27.5 nM T64765 C5O9MJ 71625826 IC50 = 0.2 nM T64765 C34MUC 71625827 IC50 = 1.4 nM T64765 CLSI36 71625828 IC50 = 0.6 nM T64765 C93WIJ 71712245 Ki = 0.2399 nM T64765 CS93OL 72164593 IC50 = 1210 nM T64765 C6P8NB 72164594 IC50 = 2840 nM T64765 C78BIH 72164719 IC50 > 10000 nM T64765 C4R3PA 72164720 IC50 > 10000 nM T64765 CF31HT 72164721 IC50 = 540 nM T64765 CXVG31 72164838 IC50 = 80 nM T64765 CMI8C2 72164839 IC50 = 180 nM T64765 CY3W8R 72164840 IC50 = 290 nM T64765 C83CTY 72164841 IC50 = 2030 nM T64765 C6MBE0 72164842 IC50 = 1040 nM T64765 C7ZWX2 72164843 IC50 = 2460 nM T64765 CTH9B6 72164844 IC50 = 4610 nM T64765 CYIO26 72164971 IC50 > 10000 nM T64765 CI5JD2 72164972 IC50 > 10000 nM T64765 CM7EX0 72164973 IC50 > 10000 nM T64765 CI8Y0V 72164974 IC50 > 10000 nM T64765 CE46KA 72375120 Ki = 1 nM T64765 CHVL93 72375121 Ki = 27 nM T64765 CB0PC5 72725528 Ki > 398.11 nM T64765 C85CSB 72725529 Ki > 10000 nM T64765 C5FN1D 72725530 Ki > 1000 nM T64765 C8BSX2 72725584 Ki = 5.012 nM T64765 CP5C9U 72725585 Ki = 0.5012 nM T64765 CC6Q5R 72771081 Ki < 100 nM T64765 CUEG26 72841751 Ki = 6.07 nM T64765 CC65OA 73213195 Ki > 10000 nM T64765 CW83DK 73213196 Ki > 10000 nM T64765 CG4V9Q 73346048 Ki = 426.58 nM T64765 C48IFJ 73346060 Ki = 0.49 nM T64765 CG8B4R 73346061 Ki = 0.64 nM T64765 C6J0TM 73346336 Ki = 2047 nM T64765 C1TC3O 73346570 IC50 = 316.23 nM T64765 CMJ6R2 73347579 Ki = 1288.25 nM T64765 C7E1KJ 73347580 Ki = 1047.13 nM T64765 C89EYU 73347592 Ki = 0.13 nM T64765 CRS97Y 73348062 IC50 = 1584.89 nM T64765 C6TLS4 73348064 IC50 = 6.31 nM T64765 CIZE25 73348065 IC50 = 125.89 nM T64765 CI3UP9 73348066 IC50 = 316.23 nM T64765 C7P5TF 73348917 IC50 = 6.5 nM T64765 C96UOF 73348918 IC50 = 0.5 nM T64765 CH89BW 73349595 IC50 = 1258.93 nM T64765 CJQ9B2 73349596 IC50 = 6309.57 nM T64765 CD7WU6 73351150 IC50 = 6.31 nM T64765 C0L9TH 73352187 Ki = 9.31 nM T64765 CO1IC6 73352624 IC50 = 15.85 nM T64765 C3CE6Q 73352625 IC50 = 1.995 nM T64765 CF3U0J 73354130 IC50 = 31.62 nM T64765 CVIH24 73354131 IC50 = 6.31 nM T64765 C4IAJ1 73354132 IC50 = 31.62 nM T64765 CH2BZ4 73355143 Ki = 707.95 nM T64765 C26IHP 73355156 Ki = 0.53 nM T64765 C1SHD7 73355647 IC50 = 79.43 nM T64765 CN8I7C 73355648 IC50 = 125.89 nM T64765 CVHQ86 73355688 Ki = 4.3 nM T64765 CS13AW 73356713 Ki = 1.212 nM T64765 CTFE46 73356714 Ki = 0.549 nM T64765 C9JBH3 73356715 Ki = 0.9 nM T64765 CE6T7X 73357178 IC50 = 19.95 nM T64765 CVR65X 73357180 IC50 = 7.943 nM T64765 C38KLR 76286162 IC50 = 2.5 nM T64765 CB2QY6 76311111 IC50 = 4.4 nM T64765 CY43DL 76311112 IC50 = 12 nM T64765 CFW19K 76311113 IC50 = 4 nM T64765 CCY14H 76314422 Ki = 4 nM T64765 C8HIS3 76314722 Ki = 0.8 nM T64765 C7K2WL 76314723 IC50 = 140 nM T64765 C1H0GX 76314724 IC50 = 2.7 nM T64765 C4R7PJ 76314725 IC50 = 18 nM T64765 CU0NR6 76314726 Ki = 3 nM T64765 CT64PM 76317221 Ki = 0.02512 nM T64765 CF9UO7 76317985 Ki = 173 nM T64765 CN8Q6E 76318296 Ki = 16 nM T64765 C4FHB2 76318297 Ki = 97 nM T64765 C1ZY4T 76318298 IC50 = 3.2 nM T64765 CRV6G8 76320902 Ki = 0.1 nM T64765 CEK3O5 76321713 EC50 = 0.5 nM T64765 CHDF36 76325614 IC50 = 1.9 nM T64765 CS27NF 76325615 Ki = 0.3 nM T64765 CI1L9C 76325616 IC50 = 21 nM T64765 C47WKY 76325617 IC50 = 340 nM T64765 CKLY67 76328872 Ki = 9.1 nM T64765 C8CQ9Y 76328873 EC50 = 0.4 nM T64765 CH9R4Y 76329180 Ki = 1670 nM T64765 C81OXN 76329181 IC50 = 0.8 nM T64765 CXI64G 76329182 IC50 = 14 nM T64765 C8H9JD 76329183 IC50 = 32 nM T64765 CAXT31 76329184 IC50 = 6.5 nM T64765 C7S0CZ 76329185 IC50 = 13 nM T64765 CL95HD 76332844 Ki > 10000000 nM T64765 CI2K3T 76332845 IC50 = 6.3 nM T64765 CT9CO2 76336463 IC50 = 1.6 nM T64765 CD7TI2 76336464 IC50 = 3.6 nM T64765 C21BOE 78320398 IC50 = 3.3 nM T64765 CV60IH 78321037 IC50 = 0.78 nM T64765 CA45JE 78321360 IC50 = 0.97 nM T64765 CL8EI6 78324474 IC50 = 8.1 nM T64765 CJ1FQ4 78324475 IC50 = 0.67 nM T64765 C1JX9C 78324476 IC50 = 5.5 nM T64765 C1GIU4 78324785 IC50 = 0.93 nM T64765 CW12TZ 78324786 IC50 = 1.2 nM T64765 CT1Y6R 78324787 IC50 = 1.1 nM T64765 CKZ8E9 78324788 IC50 = 3.1 nM T64765 C4C2RN 78324789 IC50 = 1.8 nM T64765 C35REB 86294834 Ki = 2.512 nM T64765 CSVE49 86294841 Ki = 0.4786 nM T64765 CR7Y9T 86766090 IC50 = 170 nM T64765 CG71LF 90281088 IC50 = 3.8 nM T64765 CP68KJ 90645145 Ki = 15000 nM T64765 C3U1IQ 90645147 Ki = 13200 nM T64765 CF05GE 90654501 Ki = 0.9333 nM T64765 C1BJC6 90654502 Ki = 42.66 nM T64765 CPY4X2 90654503 Ki = 75.86 nM T64765 C7W9NY 90656427 Ki = 2.951 nM T64765 CPFR56 90656428 Ki = 10.96 nM T64765 CRM9P4 90656429 Ki = 0.2291 nM T64765 C5SF0O 90666843 EC50 = 0.631 nM T64765 C8B9PX 90666844 Ki = 1.995 nM T64765 C9G8SN 90666845 Ki = 1.259 nM T64765 C52AYQ 90666846 EC50 = 1.585 nM T64765 CFA3D4 112936251 Ki = 2511.89 nM T64765 CY1BQ6 118710487 Ki = 76 nM T64765 CBT5N9 118710504 Ki = 2500 nM T64765 CU3X0M 118729231 Ki > 10000 nM T64765 CNE49D 118729233 Ki = 2 nM T64765 CLD1Z7 118729234 Ki = 2 nM T64765 C4RDW3 118729235 Ki = 4200 nM T64765 C47XHR 118729237 Ki = 2600 nM T64765 C08FQG 118729239 Ki = 680 nM T64765 CR0HA4 118729241 Ki = 5100 nM T64765 CY36XK 118729243 Ki = 230 nM T64765 C1VK9B 118729245 Ki = 1100 nM T64765 CVR67P 118729247 Ki = 530 nM T64765 CA2Y1F 118729249 Ki = 8 nM T64765 CE1IB3 118729250 Ki = 6 nM T64765 CI8WR2 118729251 Ki = 4 nM T64765 C4ML5K 118729252 Ki = 8 nM T64765 COCH98 118729253 Ki = 800 nM T64765 CQ7K5G 118729255 Ki = 1000 nM T64765 C2LDI1 118729257 Ki = 230 nM T64765 COQ04B 118729259 Ki = 4100 nM T64765 C9BG0R 118729261 Ki = 30 nM T64765 C63GWU 118729262 Ki = 60 nM T64765 CN24KA 118729263 Ki = 10 nM T64765 C7ZJ2F 118729265 Ki = 80 nM T64765 CL5W0J 118729267 Ki = 3 nM T64765 CN65HD 118729269 Ki = 94 nM T64765 C2B6YA 118729271 Ki = 430 nM T64765 CZ40RY 118729273 Ki > 10000 nM T64765 CE38GM 118729275 Ki = 200 nM T64765 CS9W7L 118729277 Ki = 60 nM T64765 C9LI7N 118729278 Ki = 190 nM T64765 C8TEX7 118729279 Ki = 120 nM T64765 CW3R9X 118729280 Ki = 400 nM T64765 CBT81N 118734854 Ki = 13 nM T64765 CT9FW8 118734855 Ki = 19 nM T64765 CRO04M 118734872 Ki = 7 nM T64765 CSYU98 118734873 Ki = 49 nM T64765 CAZP57 118734874 Ki = 39 nM T64765 C4G3YC 118734875 EC50 = 0.7 nM T64765 C9AIE1 118734876 EC50 = 0.6 nM T64765 CXZ78U 118737697 IC50 = 0.95 nM T64765 CUQ7O0 118737698 IC50 = 2.1 nM T64765 CB45KL 118737699 IC50 = 15 nM T64765 C1AVR8 118737700 IC50 = 0.99 nM T64765 CI9X7E 118737701 IC50 = 1.9 nM T64765 CU9Z3P 118737702 IC50 = 2.1 nM T64765 CX6LT1 118737703 IC50 = 1.2 nM T64765 CC3WA9 118737704 IC50 = 2.5 nM T64765 C7BFW1 118897118 Ki > 10000 nM T64765 CTBN56 127026052 Ki = 2089.3 nM T64765 CE8FB9 127035468 Ki = 1.2 nM T64765 CK1YT7 127035469 Ki = 1.8 nM T64765 CT9J7V 127035470 Ki = 0.03 nM T64765 C0Z9RT 127035835 Ki = 6025.6 nM T64765 CP0W4Y 127036068 Ki = 26.9 nM T64765 CL0AO9 127036069 Ki = 103 nM T64765 CU49VE 127036186 Ki < 10000 nM T64765 C0V4SJ 127036359 Ki = 0.9 nM T64765 CH45AM 127036360 Ki = 1 nM T64765 CGP4C1 127036361 Ki = 2.5 nM T64765 C7XL5W 127036362 Ki = 1 nM T64765 CU7C6O 127036388 Ki = 7.3 nM T64765 CS98BW 127036389 Ki = 10.5 nM T64765 CC1S9E 127036390 Ki = 11.4 nM T64765 CNGZ16 127036391 Ki = 18.4 nM T64765 CGA0L3 127036392 Ki = 7 nM T64765 C9Z2KW 127036393 Ki = 6.7 nM T64765 C5WX6V 127036558 Ki = 5.7 nM T64765 CLPS19 127036559 Ki = 9.2 nM T64765 C9QGO0 127036598 Ki = 0.1 nM T64765 CG06BD 127036932 Ki = 1584.89 nM T64765 CVW71O 127036953 Ki = 1479.11 nM T64765 C0GMJ4 127037206 Ki = 8.3 nM T64765 C7FX2E 127037207 Ki = 1.6 nM T64765 CAS36Q 127037546 Ki = 1357 nM T64765 CR7KD3 127037547 Ki = 384.3 nM T64765 C4W1ET 127038667 Ki = 800 nM T64765 CN2GQ8 127038668 Ki = 800 nM T64765 CDSN30 127038669 Ki = 371 nM T64765 CRNY45 127038670 Ki = 371 nM T64765 C7Y5PE 127038671 Ki = 255 nM T64765 C7O9LE 127038672 Ki = 174 nM T64765 C3CZ0U 127038673 Ki = 174 nM T64765 C4CN9T 127038674 Ki = 412 nM T64765 CCYM28 127038675 Ki = 412 nM T64765 CO86VY 127038676 Ki = 293 nM T64765 CA98LR 127038677 Ki = 293 nM T64765 C45PDE 127038682 Ki = 265 nM T64765 C0M2AN 127038683 Ki = 205 nM T64765 CAK7N0 127038684 Ki = 205 nM T64765 C7Z2WX 127038685 Ki = 189 nM T64765 C9VFT3 127038686 Ki = 189 nM T64765 C9W4PX 127038944 Ki = 180 nM T64765 C80CVU 127038945 Ki = 180 nM T64765 COH39R 127039026 Ki = 237 nM T64765 C9BOL2 127039027 Ki = 237 nM T64765 CK6X0N 127039028 Ki = 333 nM T64765 C1FIP3 127039029 Ki = 333 nM T64765 CLKG61 127039030 Ki = 466 nM T64765 C6TVS8 127039031 Ki = 446 nM T64765 CRJ0Z2 127039032 Ki = 805 nM T64765 CQW8E9 127039033 Ki = 805 nM T64765 CO6Q2D 127040255 Ki = 467 nM T64765 CTLX59 127040256 Ki = 467 nM T64765 CSCA42 127040266 EC50 = 72 nM T64765 C94HGO 127040267 Ki = 133 nM T64765 C9SQT3 127040591 EC50 = 75 nM T64765 C4QX1U 127040592 Ki = 128 nM T64765 CU07BR 127041243 Ki = 427 nM T64765 C6V2WB 127041329 Ki > 150000 nM T64765 CCSL97 127041626 Ki = 203 nM T64765 C9JU4M 127042151 Ki = 203 nM T64765 CXY4Q9 127042504 Ki > 150000 nM T64765 C4KO0Z 127048828 EC50 = 578 nM T64765 CY38PR 127049156 EC50 > 10000 nM T64765 CG35RK 127049855 Ki = 590 nM T64765 C5BZ6T 127049856 Ki = 745 nM T64765 CF0Y6S 127050431 EC50 = 212 nM T64765 C6F2RA 127050434 EC50 = 170 nM T64765 C5P1EB 127050776 Ki = 5680 nM T64765 CH8G4Z 127051047 Ki = 9500 nM T64765 CH8Y7R 127051301 EC50 = 370 nM T64765 C9OSN3 127052293 Ki = 1230 nM T64765 C3WA2L 127052294 Ki = 870 nM T64765 C98YAI 127052634 EC50 = 1530 nM T64765 C7T4VH 127052635 EC50 = 858 nM T64765 CS58HX 132060734 Ki = 1015 nM T64765 CY8B9L 132060743 Ki = 476.3 nM T64765 C4VNA6 132060746 Ki = 165 nM T64765 C4OC0I 132060752 Ki = 357 nM T64765 C7FM0U 132060763 Ki = 2791 nM T64765 CT81OY 132060776 Ki = 300 nM T64765 CAVB41 132584404 Ki > 10000 nM T64765 CUFQ23 134132637 Ki = 34 nM T64765 CQ95LB 134133571 Ki = 1.585 nM T64765 CG9J7V 134136763 Ki = 0.631 nM T64765 C3W5SM 134139893 Ki = 0.3981 nM T64765 CHG9Z5 134140686 Ki = 1.995 nM T64765 CFW7E3 134141385 Ki = 1.259 nM T64765 C3NT1H 134143679 Ki = 0.5012 nM T64765 C2IM4X 134143913 Ki = 3.162 nM T64765 CBU81N 134149168 Ki = 814 nM T64765 C1PQ5T 134150412 Ki = 1.585 nM T64765 CUD08L 134817200 Ki = 10.8 nM T64765 CHSN19 135525668 Ki = 3090 nM T64765 CU57CI 135887269 Ki = 192 nM T64765 C5KE3N 135986088 Ki = 3.27 nM T64765 CBS93O 136030655 Ki > 10000 nM T64765 CFC17Q 136042268 Ki = 1190 nM T64765 CN5B6D 136042269 Ki > 20000 nM T64765 CH9J5X 136042270 Ki = 3810 nM T64765 CAQZ86 136042385 Ki = 153 nM T64765 CMD9J0 136097741 Ki = 213 nM T64765 C8I7CO 136141537 Ki > 10000 nM T64765 CRH19Y 136192874 Ki > 10000 nM T64765 C56FVS 136192886 Ki = 2511.89 nM T64765 CI8NR9 137632569 Ki = 14 nM T64765 C4XEF0 137634349 Ki = 22 nM T64765 CPCY48 137645406 Ki = 509 nM T64765 C7CM5W 137655927 Ki = 258 nM T64765 CWO0B6 137657169 Ki = 9.6 nM T64765 C8M2UW 137659490 Ki = 47 nM T64765 CT7R5X 145949589 EC50 = 0.1 nM T64765 C0H1AE 145949735 Ki = 16 nM T64765 CJ7I6M 145949790 Ki = 683 nM T64765 CQV3H0 145950629 Ki > 10000 nM T64765 CJ1T8Q 145950879 Ki > 10000 nM T64765 C9LA5R 145950903 Ki > 10000 nM T64765 CE1VU8 145951024 Ki = 3654 nM T64765 C2QK7V 145951081 EC50 = 3.8 nM T64765 C8SV0W 145951662 Ki = 8740 nM T64765 C8X4CL 145951678 EC50 = 10 nM T64765 C0CFI7 145951910 Ki > 10000 nM T64765 CM13ID 145951920 EC50 = 24 nM T64765 CN87EM 145952154 Ki = 5405 nM T64765 C49UCV 145952531 EC50 = 186.21 nM T64765 CR4G5B 145952665 EC50 = 3 nM T64765 CK29XC 145952741 EC50 = 61.66 nM T64765 CI5OT6 145953540 Ki = 30.6 nM T64765 CFSC86 145953579 EC50 = 104 nM T64765 C8TJU1 145954176 EC50 = 14.4 nM T64765 C5V4GU 145954498 EC50 = 1.23 nM T64765 CY1Z6C 145954511 Ki = 3827 nM T64765 CCH60G 145954725 EC50 = 2.692 nM T64765 C53CQS 145954741 EC50 = 93.33 nM T64765 CKT86N 145955209 Ki = 883 nM T64765 C49YFS 145955462 Ki = 6212 nM T64765 C20OFI 145955602 Ki = 3420 nM T64765 CF2GK0 145956355 EC50 = 0.263 nM T64765 CCX97Y 145956362 EC50 = 0.1 nM T64765 CYM7W1 145956417 Ki = 120 nM T64765 CNBG57 145956619 Ki > 10000 nM T64765 CQFK74 145956781 EC50 = 1.1 nM T64765 CHOV56 145956810 Ki = 8156 nM T64765 C0EKG9 145956832 Ki = 482 nM T64765 CB6A2O 145957226 EC50 = 13 nM T64765 CN2HX4 145958231 Ki = 37.8 nM T64765 CXN73I 145958342 Ki = 5477 nM T64765 C0VF1M 145958501 Ki = 2264 nM T64765 C6QBR4 145958654 Ki > 10000 nM T64765 CWF29C 145959270 Ki = 2957 nM T64765 CF01LC 145959298 EC50 = 1.288 nM T64765 C2O9NR 145960088 Ki = 5196 nM T64765 CLA7K6 145960431 Ki = 43.3 nM T64765 C9Z8WS 145961016 Ki = 21 nM T64765 C8W1VL 145961232 Ki = 32.8 nM T64765 C67GQI 145961372 Ki = 21.9 nM T64765 CJ80QU 145961549 Ki = 55.9 nM T64765 CON7E1 145961579 Ki = 126 nM T64765 CI7MT0 145961606 Ki = 5.4 nM T64765 C09JYK 145961641 EC50 = 6.607 nM T64765 CQS1G2 145961721 Ki = 69.3 nM T64765 C3A7OI 145961804 Ki = 95 nM T64765 CV06SC 145962308 Ki = 42.3 nM T64765 CHQF93 145962776 Ki = 47.6 nM T64765 C8DV1J 145962869 Ki = 57.3 nM T64765 CJZO20 145963266 Ki = 69 nM T64765 CPX2M3 145963301 Ki = 92.1 nM T64765 CIAD71 145964098 IC50 > 30000 nM T64765 C6TF7H 145964274 Ki = 2.1 nM T64765 CS51VC 145966675 IC50 = 2600 nM T64765 CG78KQ 145967442 Ki = 3.9 nM T64765 CS47PW 145967736 Ki = 182.5 nM T64765 CKY53A 145967933 Ki = 60.5 nM T64765 CCH2J8 145968136 Ki = 46.5 nM T64765 CWT5X8 145968175 Ki = 8.8 nM T64765 CI17YH 145968353 Ki = 238 nM T64765 C1XI5A 145968394 Ki = 128.3 nM T64765 C8Z3HO 145968893 Ki = 120.7 nM T64765 C0CU8H 145969075 Ki = 325.9 nM T64765 C8X0AR 145969247 Ki = 36.6 nM T64765 CM3BL4 145969287 Ki = 41.2 nM T64765 CL1I2F 145969682 Ki = 13.6 nM T64765 CCG3K6 145969758 Ki = 308.1 nM T64765 CKI8J2 145969780 Ki = 64.4 nM T64765 CN2OA7 145969926 Ki = 33.8 nM T64765 CW8K4O 145969939 Ki = 21.4 nM T64765 CGSV09 145970236 Ki = 55 nM T64765 CQ52DS 145970357 Ki = 68 nM T64765 C97VSH 145971024 Ki = 2.2 nM T64765 C5FT7K 145971137 Ki = 23.4 nM T64765 CH31NI 145971293 EC50 = 0.2692 nM T64765 C2EV1M 145971387 Ki = 696 nM T64765 C20HME 145973591 EC50 = 2.7 nM T64765 CT5CX0 145973771 Ki = 2770 nM T64765 C3J7YA 145973881 Ki = 11 nM T64765 C0OCN5 145973963 Ki = 39 nM T64765 CYRO78 145974564 EC50 = 5.623 nM T64765 CU15SA 145974947 Ki = 32 nM T64765 C79AKX 145975223 Ki = 304 nM T64765 C9ME5T 145975612 IC50 = 280 nM T64765 C8BOR1 145977335 Ki = 33 nM T64765 C8IAL2 145977624 Ki = 6.5 nM T64765 CB4E3T 145982627 Ki = 1600 nM T64765 CYH8L5 145982763 Ki = 54 nM T64765 CO52DH 145982869 Ki = 87 nM T64765 C96EKT 145982899 Ki = 930 nM T64765 CJW17E 145982964 Ki = 72 nM T64765 CDO8T7 145983010 Ki = 98 nM T64765 CK6O5E 145983057 Ki = 22 nM T64765 C28FQJ 145983140 Ki = 130 nM T64765 CLVA73 145983142 Ki > 5000 nM T64765 CBC0V2 145983174 Ki > 5000 nM T64765 CPX5M3 145983216 Ki = 220 nM T64765 CB9H3V 145983280 Ki = 125.89 nM T64765 CDJ8V4 145983293 Ki > 5000 nM T64765 CFEA75 145983320 Ki = 1100 nM T64765 C2TE4K 145983486 Ki = 1600 nM T64765 C0WD8T 145983501 Ki = 450 nM T64765 CN3LD5 145983517 Ki = 190 nM T64765 C48KYO 145983584 Ki = 450 nM T64765 C6KXI0 145983609 Ki = 21 nM T64765 CE5Z7O 145983713 Ki = 47 nM T64765 CZEN06 145983723 Ki = 5800 nM T64765 CZV1R3 145983822 Ki = 57 nM T64765 CP71OV 145983845 Ki = 200 nM T64765 C8CA7J 145983990 Ki = 4.2 nM T64765 C3L5OY 145984019 Ki = 380 nM T64765 C8FMY2 145984071 Ki = 7 nM T64765 CN9GM2 145984096 Ki = 1300 nM T64765 C6U3IB 145984317 Ki = 44 nM T64765 CWOF31 145984339 Ki = 170 nM T64765 CFQ5O0 145984448 Ki = 100 nM T64765 C2M5PV 145984454 Ki > 10000 nM T64765 CVDN71 145984498 Ki > 5000 nM T64765 C5CI7Z 145984562 Ki = 410 nM T64765 CBP9F4 145984670 Ki = 600 nM T64765 CY01AF 145984758 Ki = 110 nM T64765 CXDP23 145984763 Ki = 280 nM T64765 CP1LA9 145984809 Ki = 2000 nM T64765 C03QVW 145984823 Ki = 430 nM T64765 CN6KP4 145984963 Ki = 1300 nM T64765 C50AYD 145984996 Ki = 300 nM T64765 C8Q5IR 145985024 Ki = 5700 nM T64765 C6XE8C 145985206 Ki = 4100 nM T64765 C6AXO9 145985222 Ki = 5.4 nM T64765 CEYS38 145985247 Ki = 147.91 nM T64765 CTD4Q2 145985274 Ki = 42 nM T64765 CUS59J 145985351 Ki > 5000 nM T64765 C4ALN8 145985452 Ki = 200 nM T64765 CMLS93 145985490 Ki = 1071.52 nM T64765 C41RQV 145985537 Ki > 5000 nM T64765 CT52FI 145985559 Ki > 5000 nM T64765 CHZL14 145985673 Ki > 5000 nM T64765 CHC87W 145985703 Ki = 489.78 nM T64765 C8XH4Z 145985731 Ki > 5000 nM T64765 CC9OQ3 145985775 Ki = 2100 nM T64765 CHY4F5 145985790 Ki = 520 nM T64765 CJ3QF9 145985902 Ki = 5900 nM T64765 C70QAR 145986049 Ki = 1100 nM T64765 C1OM3W 145986109 Ki = 870 nM T64765 CDY73H 145986572 Ki = 46 nM T64765 CV9G7Z 153287572 Ki > 10000 nM T64765 CO85KL 153287574 Ki = 3981.07 nM T64765 C51NYU 155510452 Ki = 157 nM T64765 C5U8JC 155510520 IC50 > 50000 nM T64765 CRI91T 155511196 Ki = 437 nM T64765 CLC7N6 155511939 Ki = 42 nM T64765 CR8M5G 155512115 Ki > 1000 nM T64765 CHD1Y5 155512264 Ki = 115 nM T64765 CGAP59 155512724 Ki = 5623.41 nM T64765 CL3D0I 155513598 IC50 > 10000 nM T64765 C20UBG 155513611 Ki = 144.54 nM T64765 CN5VE4 155513723 Ki = 317 nM T64765 C6OLV9 155513736 Ki = 100 nM T64765 CO98BH 155513780 Ki = 2.6 nM T64765 C37HQI 155513820 IC50 = 730 nM T64765 COIR08 155514045 Ki = 6.4 nM T64765 CG7P9N 155514324 Ki = 9.51 nM T64765 CSCV74 155514975 Ki = 10.8 nM T64765 CMZ4Q7 155515478 EC50 = 0.3162 nM T64765 CNLU19 155515879 Ki = 212.1 nM T64765 CTZL14 155516421 Ki = 27.54 nM T64765 C14CHU 155516491 Ki > 10000 nM T64765 CTR7C8 155516568 Ki = 60 nM T64765 CAW29B 155517379 Ki = 18 nM T64765 C7Y8RB 155517663 Ki = 22.1 nM T64765 CGO36Z 155517879 Ki = 1122.02 nM T64765 CC01KR 155517939 Ki = 1720 nM T64765 CY07UN 155517942 Ki = 1.1 nM T64765 CVQS21 155518359 Ki = 22 nM T64765 C2UOV4 155518892 Ki = 5.6 nM T64765 CVUJ59 155519557 IC50 = 5495.41 nM T64765 CZ8L7H 155519671 Ki = 377 nM T64765 CE2YP0 155520226 Ki = 690 nM T64765 C9Q5XZ 155520394 Ki = 3572 nM T64765 C2GAV1 155520534 Ki = 140 nM T64765 CY7T3U 155521079 IC50 > 50000 nM T64765 C8FIB1 155521219 Ki = 5.2 nM T64765 CT0QF1 155521380 Ki = 89 nM T64765 CY2CK4 155521688 Ki = 0.6 nM T64765 CM4TF8 155522043 Ki = 31 nM T64765 C13NYD 155522219 IC50 = 40 nM T64765 C10YAR 155522254 Ki = 2.8 nM T64765 C9JL5R 155522294 Ki = 4040 nM T64765 CKRY85 155522812 Ki = 499 nM T64765 CM5LN9 155522957 Ki = 3697 nM T64765 C50XJS 155523039 Ki = 3390 nM T64765 C7Y6LX 155523256 IC50 = 66.07 nM T64765 CHD0W2 155523356 Ki = 915 nM T64765 CW5F4L 155523500 Ki = 181.5 nM T64765 CI2Z8F 155524114 Ki = 3.311 nM T64765 C2SLK7 155524693 EC50 = 3.981 nM T64765 CA9GL1 155524804 Ki = 1.61 nM T64765 CWE2B5 155524877 Ki = 159.8 nM T64765 C56QGZ 155524883 Ki = 83 nM T64765 CQS1N5 155525278 Ki = 13.8 nM T64765 C2K4YP 155525816 IC50 = 549.54 nM T64765 C7L2KF 155526307 Ki > 1000 nM T64765 C0ZBJ1 155526345 EC50 = 5.012 nM T64765 CUS6X0 155527111 Ki = 50.12 nM T64765 C13TUC 155527319 EC50 = 31.62 nM T64765 C72JHU 155528281 Ki = 234 nM T64765 C06FHD 155528291 EC50 = 63.1 nM T64765 C5JZ6K 155529212 Ki = 115 nM T64765 CSX93I 155529365 IC50 = 12.8 nM T64765 CJO4C6 155529822 IC50 = 3090.3 nM T64765 C08UZD 155529825 Ki = 0.7 nM T64765 C1FW0Q 155530764 Ki = 1444 nM T64765 CR52CO 155530956 Ki > 1000 nM T64765 C3CPQ2 155531145 Ki = 6 nM T64765 CR9S6W 155531303 Ki = 159 nM T64765 CD4F1G 155531771 Ki > 10000 nM T64765 C3F1PE 155531878 Ki = 266 nM T64765 C1NQD7 155532178 EC50 = 1.259 nM T64765 CC6ZE7 155532308 Ki = 1230 nM T64765 CEB3I8 155532429 Ki = 1392 nM T64765 CCA9G7 155532528 Ki = 260 nM T64765 C1E5FH 155532722 IC50 = 2930 nM T64765 CF9V4T 155533283 Ki = 3.2 nM T64765 CF7Z8V 155533291 EC50 = 15.85 nM T64765 C56BHV 155533413 Ki = 40 nM T64765 CYFL52 155533425 EC50 = 10 nM T64765 C80YPT 155533743 Ki = 92 nM T64765 CRBU15 155533940 EC50 = 12.59 nM T64765 CR70SX 155533943 Ki > 1000 nM T64765 C74TAG 155534484 Ki = 9.5 nM T64765 C8XG9P 155534518 Ki = 9.333 nM T64765 CV83SG 155534733 Ki = 4520 nM T64765 CJH0I7 155534759 Ki = 1.9 nM T64765 CH2S1W 155534883 IC50 > 50000 nM T64765 CNK51Q 155535097 Ki > 10000 nM T64765 CGXM42 155535113 Ki = 3627 nM T64765 CC9J6W 155535840 Ki > 1000 nM T64765 CB79ZW 155536080 Ki > 10000 nM T64765 C17MFJ 155536277 Ki = 908 nM T64765 CLG47F 155536506 Ki = 147 nM T64765 CRI5F4 155536508 Ki = 9.55 nM T64765 C6C5NV 155536937 Ki = 228.2 nM T64765 CG6P2Z 155537026 Ki = 30 nM T64765 CBT38O 155537566 Ki = 60 nM T64765 CMP4H0 155537748 Ki = 1.07 nM T64765 CCB1A2 155537946 Ki > 1000 nM T64765 CQ02MZ 155538072 Ki > 1000 nM T64765 CM9VU3 155538173 Ki = 30 nM T64765 CV1F2G 155538221 EC50 = 3.162 nM T64765 CYA2O8 155538400 Ki = 374 nM T64765 CIS8K6 155538406 Ki = 3.3 nM T64765 CC42BH 155538520 Ki = 3.8 nM T64765 C9I2CK 155538966 IC50 = 4610 nM T64765 C6QN1S 155538988 Ki = 3467.37 nM T64765 CI37OT 155539096 Ki > 10000 nM T64765 C3YW8J 155539458 Ki = 501.19 nM T64765 C37JBM 155539543 Ki = 122 nM T64765 C7YD2U 155539915 Ki = 11 nM T64765 CN20LJ 155540111 IC50 = 520 nM T64765 CK1G0I 155540170 Ki = 9 nM T64765 COF72J 155540201 Ki = 275.42 nM T64765 CR6M9Y 155540792 EC50 = 1.995 nM T64765 CHQ7A8 155541279 Ki = 537.03 nM T64765 CQ5YB9 155541512 Ki = 1.9 nM T64765 CT6UN1 155541545 Ki = 1619 nM T64765 CKI4P5 155541610 Ki = 111 nM T64765 C4GO2A 155541779 Ki = 2316 nM T64765 CTO07F 155541808 Ki = 395 nM T64765 C2HJ4K 155541911 EC50 = 100 nM T64765 C96YSN 155542256 IC50 = 4450 nM T64765 C8IV6K 155542570 Ki = 9.17 nM T64765 CKTW02 155543125 Ki = 532.1 nM T64765 CDO05U 155543223 Ki = 580 nM T64765 CC4KN9 155543685 Ki = 298 nM T64765 CTN6Y0 155543865 Ki = 1634 nM T64765 CIEQ43 155543869 Ki = 344 nM T64765 CZT91D 155543973 Ki = 848 nM T64765 C1OG6N 155544052 Ki = 35 nM T64765 CBK4I2 155544071 IC50 = 2691.53 nM T64765 CP1FI5 155544094 Ki = 1392 nM T64765 C1F9ZD 155544305 Ki = 34 nM T64765 CGFI39 155544432 EC50 = 7.943 nM T64765 CBH39J 155544597 Ki = 5 nM T64765 CI5HT7 155544816 IC50 = 4680 nM T64765 C5EV7C 155544839 IC50 = 12300 nM T64765 CNQ0F4 155544914 Ki = 425 nM T64765 CK9T1E 155545703 Ki = 84.3 nM T64765 CAY2P0 155545717 Ki = 186 nM T64765 CVF2T8 155545893 Ki = 753 nM T64765 CJBP49 155546194 Ki = 299 nM T64765 CO2J0Z 155546798 Ki = 5495.41 nM T64765 C3G9OU 155547176 Ki = 192 nM T64765 CO3GW7 155547596 Ki = 2.6 nM T64765 CDG54R 155547601 EC50 = 0.631 nM T64765 C46OZR 155548338 IC50 = 6760.83 nM T64765 C1T0BF 155549318 Ki = 3019.95 nM T64765 CF21PW 155549506 Ki = 9 nM T64765 C29BAV 155550731 IC50 = 4.04 nM T64765 CPMR12 155551283 Ki > 1000 nM T64765 CDE3P0 155551319 Ki = 4889 nM T64765 CT1I9G 155551737 Ki = 23.6 nM T64765 C7WO9P 155552060 Ki = 2398.83 nM T64765 CZQW48 155552101 Ki = 6025.6 nM T64765 CLK7U1 155552340 Ki = 204.17 nM T64765 C7DM5X 155552772 Ki > 1000 nM T64765 CV9SY1 155552989 Ki = 294 nM T64765 C8BVH4 155553066 Ki = 26 nM T64765 CR62OS 155553226 Ki > 10000 nM T64765 C1RLI0 155553370 Ki = 2.6 nM T64765 C4ERQ3 155553614 Ki = 10.2 nM T64765 C1LIT7 155553731 Ki = 10.4 nM T64765 CE9T1I 155553838 Ki = 2.9 nM T64765 CMD3T6 155553964 IC50 = 900 nM T64765 C0F2DU 155554431 Ki > 1000 nM T64765 CA6T8X 155554941 Ki > 1000 nM T64765 CZ01CH 155555041 Ki = 15.8 nM T64765 CP5XO6 155555134 Ki > 10000 nM T64765 CTYU50 155555523 IC50 = 410 nM T64765 CQ8I3X 155555700 IC50 = 1940 nM T64765 CVQ6O4 155555986 Ki = 83 nM T64765 C13XWK 155556196 Ki = 10 nM T64765 C5VKG2 155556251 Ki = 151 nM T64765 C5BEX2 155556301 Ki = 11.7 nM T64765 CJ75TC 155556370 Ki = 6.7 nM T64765 C03CHA 155556460 IC50 = 430 nM T64765 CXI70N 155556709 IC50 > 50000 nM T64765 CJR39N 155557368 EC50 = 7.943 nM T64765 C6Q2YJ 155558288 Ki = 54 nM T64765 CP1HC2 155558360 EC50 = 0.7943 nM T64765 CJT90H 155558487 Ki = 6 nM T64765 C2VI9G 155558502 Ki = 100 nM T64765 CP71KI 155558614 Ki = 522.8 nM T64765 C0YIQ1 155558898 Ki = 63 nM T64765 CGH2Y1 155559319 IC50 = 1288.25 nM T64765 C5BAG2 155559502 Ki > 10000 nM T64765 CM9B8P 155559800 Ki = 8.3 nM T64765 C06BZW 155559811 Ki = 280 nM T64765 C3XO6J 155560605 IC50 = 270 nM T64765 C57DRK 155560636 Ki = 18 nM T64765 CJ9R1T 155561102 Ki = 214 nM T64765 C07DYC 155561219 Ki = 302 nM T64765 C54MEX 155561493 Ki = 1455 nM T64765 C4V2TY 155561504 Ki = 315 nM T64765 CEN7Q6 155562440 EC50 = 31.62 nM T64765 CFHB16 155562868 Ki = 107.6 nM T64765 CJ2S0E 155563066 Ki = 121 nM T64765 CJQ59S 155563181 Ki = 565 nM T64765 CLC7W8 155563295 Ki = 7 nM T64765 C9S7PB 155564518 Ki = 2.4 nM T64765 C9N5VK 155564956 Ki = 4.8 nM T64765 CCM3U6 155565090 Ki = 2453 nM T64765 C1IHS2 155565227 Ki = 4.49 nM T64765 C4H3WJ 155565266 Ki = 2 nM T64765 CEK58B 155565576 EC50 = 5.012 nM T64765 CW9K2D 155565634 EC50 = 39.81 nM T64765 C9DMO1 155565722 Ki = 1.5 nM T64765 CQ75DA 155565842 IC50 = 90 nM T64765 CWEU60 155566502 IC50 = 2070 nM T64765 C7ZUE1 155566557 Ki = 1.2 nM T64765 C8HR4Q 155567029 IC50 = 9.08 nM T64765 C8KY4O 155567055 Ki > 1000 nM T64765 CW0VX4 155567092 Ki = 76 nM T64765 CHD6C8 155567107 Ki = 691.83 nM T64765 CL54XY 155567151 IC50 = 240 nM T64765 CCR6S2 155567442 Ki = 448 nM T64765 C6I5QA 155567666 Ki = 317 nM T64765 C8M3OG 155567862 Ki = 25.4 nM T64765 C5G3FT 155568977 Ki = 52 nM T64765 C19LOV 155569239 Ki = 15.4 nM T64765 C7SH2R 155569586 Ki = 0.96 nM T64765 C3N9VU 10251906 Ki > 500 nM T64765 CP9TR0 10324985 Ki > 10000 nM T64765 CB0I4L 24884859 Ki = 0.1585 nM T64765 C7Y0EQ 24885255 Ki = 1 nM T64765 CYV2S9 24885661 Ki = 2.512 nM T64765 C5Z2KD 24886136 Ki = 0.3162 nM T64765 CS5N4V 24886137 Ki = 1.995 nM T64765 CP2O0E 24886138 Ki = 2.512 nM T64765 CZO3R2 24886366 Ki = 5.012 nM T64765 C90ROZ 24886368 Ki = 1.585 nM T64765 C7BYA1 44254046 Ki = 0.631 nM T64765 C65JLI 44254219 Ki = 6.31 nM T64765 D00AWM 9826520 Ki = 208 nM T64765 D00HWF 6421522 Ki = 2.512 nM T64765 D00IIQ 44456366 Ki = 20 nM T64765 D00SHX 44456331 Ki = 400 nM T64765 D00XJR 10446295 EC50 = 3162.28 nM T64765 D01CJZ 10330240 Ki = 4.467 nM T64765 D01DAU 24825518 Ki = 3.162 nM T64765 D01JXM 46222048 Ki = 0.17 nM T64765 D01RTR 44455920 Ki = 300 nM T64765 D01XZI 10015055 Ki = 30 nM T64765 D02BXA 238317 Ki > 350 nM T64765 D02HNE 44456451 Ki = 190 nM T64765 D02IJW 44456500 Ki = 140 nM T64765 D02INJ 46222042 Ki = 56 nM T64765 D02RAN 3692 EC50 = 0.1259 nM T64765 D02SQF 37463 Ki = 6309.57 nM T64765 D03QGB 2766326 Ki = 0.2 nM T64765 D03SAM 156615 EC50 = 0.3162 nM T64765 D04FUZ 44582620 Ki = 62 nM T64765 D04LFK 44456057 Ki = 219 nM T64765 D04MKB 46898078 Ki = 11.2 nM T64765 D04NWI 44456132 Ki = 5 nM T64765 D05ANV 44456128 Ki = 81 nM T64765 D05BYD 9906860 Ki = 758.58 nM T64765 D05JZQ 44456361 Ki = 270 nM T64765 D05OHN 12226582 Ki = 4800 nM T64765 D05PBN 44456127 Ki = 5 nM T64765 D05RGW 11313837 EC50 = 0.3162 nM T64765 D05ZUX 44207909 Ki >= 1000 nM T64765 D06KLQ 44403742 Ki = 10.6 nM T64765 D06MGO 44456094 Ki = 31 nM T64765 D06NXK 46890563 Ki = 7.4 nM T64765 D06RNM 3032915 Ki = 84 nM T64765 D06RPY 11314275 Ki = 2.9 nM T64765 D07LCM 18365007 Ki = 260 nM T64765 D07PSG 52946272 Ki = 63 nM T64765 D07TST 12647300 Ki = 1600 nM T64765 D07UCE 44563685 Ki = 326 nM T64765 D08BSG 132937 EC50 = 0.05012 nM T64765 D08DOG 25130235 Ki = 1288.25 nM T64765 D08ECP 912 EC50 = 0.3981 nM T64765 D09JSA 9903343 Ki = 3.1 nM T64765 D09ROG 2994072 Ki = 11 nM T64765 D09RPR 16737207 Ki > 10000 nM T64765 D09WQL 9989505 EC50 = 0.1585 nM T64765 D0A4XL 3614 Ki = 20000 nM T64765 D0A9QT 44456154 Ki = 10.6 nM T64765 D0B4SF 41376 Ki = 67 nM T64765 D0B5SF 46222044 Ki = 9.9 nM T64765 D0B6CA 238432 Ki = 350 nM T64765 D0BI4T 53315878 Ki = 45 nM T64765 D0C1LI 53378764 Ki = 84.2 nM T64765 D0C8IB 10680721 Ki = 12 nM T64765 D0CI9W 11452311 Ki = 0.1259 nM T64765 D0D0FV 44455953 Ki = 200 nM T64765 D0D9JL 44456174 Ki = 200 nM T64765 D0DC1P 44592097 Ki = 43 nM T64765 D0E5EB 9793868 EC50 = 2.344 nM T64765 D0E5XM 13499360 EC50 = 0.631 nM T64765 D0E9SR 4908365 EC50 = 1000 nM T64765 D0F2XZ 44455952 Ki = 340 nM T64765 D0FF0Z 24825516 Ki = 1.82 nM T64765 D0FK6T 11337173 Ki = 28 nM T64765 D0FN7I 44407803 Ki = 6 nM T64765 D0G2BS 5013 Ki = 410 nM T64765 D0G5DU 44563683 Ki = 249 nM T64765 D0G5TD 44456090 Ki = 65 nM T64765 D0H2KD 921599 Ki = 9000 nM T64765 D0H3DY 10374457 EC50 = 5.888 nM T64765 D0H3LF 11393294 Ki = 6.8 nM T64765 D0H4ID 10489384 Ki = 31 nM T64765 D0H4TP 9798547 Ki = 0.12 nM T64765 D0H9IH 44456091 Ki = 16 nM T64765 D0HF4I 46888007 Ki = 24 nM T64765 D0I3XA 6422124 Ki = 46 nM T64765 D0I4BC 44455950 Ki = 30 nM T64765 D0I4UU 9990388 Ki = 2.1 nM T64765 D0J6NI 49799252 Ki = 30 nM T64765 D0J6XO 9884746 Ki = 2.754 nM T64765 D0K7XM 362025 Ki = 30 nM T64765 D0K8DZ 11672774 Ki = 15.85 nM T64765 D0K9WJ 11324846 Ki = 13 nM T64765 D0KK4C 10154137 Ki = 1.3 nM T64765 D0L5MW 181743 Ki > 10000 nM T64765 D0M2HC 46222043 Ki = 14 nM T64765 D0M7QR 44456496 Ki = 230 nM T64765 D0M9IC 441082 Ki = 3.467 nM T64765 D0MP8E 3063228 Ki = 316.23 nM T64765 D0MR0Z 44456056 Ki = 2.3 nM T64765 D0MX0Z 44456330 Ki = 21 nM T64765 D0N3OH 10389213 Ki = 93 nM T64765 D0N6CB 52940790 Ki = 20 nM T64765 D0N7KK 44456023 Ki = 230 nM T64765 D0O3GR 10681081 Ki = 47 nM T64765 D0O9YL 44456095 Ki = 35 nM T64765 D0OB7B 45482707 Ki = 139 nM T64765 D0OM9G 3035842 EC50 = 0.03981 nM T64765 D0P2UM 18071365 Ki = 2 nM T64765 D0P8SU 23635021 Ki = 96 nM T64765 D0P8UI 44456126 Ki = 27 nM T64765 D0PC7A 10106214 Ki = 2 nM T64765 D0Q0YC 11370427 Ki = 6 nM T64765 D0Q8BS 6603865 EC50 = 10 nM T64765 D0Q8CE 46222046 Ki = 2.2 nM T64765 D0Q8LU 45482781 Ki = 128 nM T64765 D0Q8NO 10176414 EC50 = 0.5012 nM T64765 D0QP3A 44455916 Ki = 5 nM T64765 D0R2TU 10774476 Ki = 27 nM T64765 D0RP8X 9925627 Ki = 39 nM T64765 D0S0HT 9812843 EC50 = 38.9 nM T64765 D0S5ON 10536901 Ki = 360 nM T64765 D0S5VI 40012125 Ki = 94 nM T64765 D0SQ0T 10942498 EC50 > 0.0001 nM T64765 D0T2RY 9948320 Ki >= 1000 nM T64765 D0T5KC 44456332 Ki = 96 nM T64765 D0T8MV 44456055 Ki = 8.9 nM T64765 D0T8OD 2790 Ki = 0.3388 nM T64765 D0TW9N 12226576 Ki = 9000 nM T64765 D0U1DR 11492393 Ki = 10 nM T64765 D0UK0F 753256 Ki = 1080 nM T64765 D0UO2Z 46222047 Ki = 4.1 nM T64765 D0UW9I 44456131 Ki = 32 nM T64765 D0V9AJ 23061353 Ki = 340 nM T64765 D0W2HJ 17805318 Ki = 41 nM T64765 D0W7OR 9877454 Ki = 588.84 nM T64765 D0X5DB 46222045 Ki = 0.89 nM T64765 D0X6SR 44456501 Ki = 70 nM T64765 D0Y5WD 44592096 Ki = 17.3 nM T64765 D0ZY8V 44563684 Ki = 274 nM T02728 D0G0TS 119192 IC50 = 82 nM T02728 D0LI1C 44469321 IC50 > 10000 nM T02728 CA74VF 4308 EC50 = 216 nM T02728 C7A3EH 1230851 EC50 = 26000 nM T02728 CA1Y2P 1230852 EC50 = 5900 nM T02728 C7L1HF 1920221 EC50 > 80000 nM T02728 C4G9CE 1941471 EC50 > 80000 nM T02728 C3P9EW 1951822 EC50 > 80000 nM T02728 C20LJC 4679731 EC50 = 20000 nM T02728 C31MKE 10056201 Ki = 190 nM T02728 CA95RS 10259186 IC50 = 3.9 nM T02728 CQR16D 10339735 EC50 > 80000 nM T02728 CYA4F6 10349413 IC50 = 19 nM T02728 C8ONE5 10418825 IC50 = 0.4 nM T02728 CU1N7K 10440485 Ki = 95 nM T02728 CD6YQ3 10463386 Ki = 3500 nM T02728 CD7V5K 10866193 IC50 = 2.5 nM T02728 CP6F2G 10931321 IC50 = 0.3 nM T02728 CSG31T 10953372 IC50 = 10.2 nM T02728 CUMK12 10953373 IC50 = 0.6 nM T02728 C0RFD9 11018748 IC50 = 106 nM T02728 C5ZFG1 11040576 IC50 = 0.3 nM T02728 C96MIU 11051535 IC50 = 6.3 nM T02728 CT87MR 11062253 IC50 = 24.6 nM T02728 CNPH25 11126117 IC50 = 0.4 nM T02728 CF04UG 11228237 Ki = 17000 nM T02728 CX0E6T 11285912 Ki = 12 nM T02728 CO47VD 11657884 IC50 = 5.71 nM T02728 CX1KQ9 11768458 IC50 = 0.5 nM T02728 CT01PL 15513866 IC50 = 1 nM T02728 CCZ40B 16114081 EC50 = 178 nM T02728 C9KCA5 24868215 IC50 = 0.33 nM T02728 CHS59N 25077380 IC50 = 22.1 nM T02728 C5LVD4 44123840 EC50 = 1.4 nM T02728 CFP9S1 44157038 EC50 = 67 nM T02728 CXV65L 44157039 EC50 = 986 nM T02728 C4P9JG 44157040 EC50 = 220 nM T02728 CWH45F 44157044 EC50 = 1214 nM T02728 CQJ03K 44342663 IC50 > 1000 nM T02728 CWF94S 44342966 IC50 = 21.7 nM T02728 C37KMX 44342967 IC50 = 11.87 nM T02728 C61OFG 44342968 IC50 = 42.4 nM T02728 CS64NI 44354075 IC50 = 0.38 nM T02728 CWJX37 44354085 IC50 = 0.4 nM T02728 C0J9UW 44354086 IC50 = 1.2 nM T02728 C5Y7PD 44354087 IC50 = 0.3 nM T02728 COFV37 44354088 IC50 = 0.25 nM T02728 C5F9XB 44354111 IC50 = 0.4 nM T02728 CP9TU5 44354112 IC50 = 0.52 nM T02728 CE7C0O 44354113 IC50 = 0.28 nM T02728 C3LE1I 44354120 IC50 = 0.4 nM T02728 C3SAZ7 44354121 IC50 = 133 nM T02728 CR82IU 44354154 IC50 = 0.34 nM T02728 CJL69G 44354211 IC50 = 0.51 nM T02728 C51YEP 44354212 IC50 = 0.34 nM T02728 CTW49H 44354244 IC50 = 0.3 nM T02728 C96DTU 44354245 IC50 = 0.3 nM T02728 C7UL8I 44354302 IC50 = 0.36 nM T02728 C39YIP 44354303 IC50 = 0.24 nM T02728 CH8W9B 44354304 IC50 = 0.59 nM T02728 CU0SY5 44354305 IC50 = 1.6 nM T02728 C1GH3Q 44360189 IC50 = 14.7 nM T02728 CSY62F 44360217 IC50 = 8.8 nM T02728 CNS8P9 44360330 IC50 = 9.3 nM T02728 C0VP5A 44360331 IC50 = 1.3 nM T02728 C8XQW1 44360527 IC50 = 28 nM T02728 CK05WA 44363448 Ki = 1.81 nM T02728 CNK7H5 44363934 Ki = 0.14 nM T02728 C2H1UE 44384829 Ki = 100 nM T02728 C9VG7J 44387547 IC50 = 11.5 nM T02728 C2APH8 44387548 IC50 = 113 nM T02728 C28DWP 44396910 Ki > 100000 nM T02728 COX1L7 44396911 Ki = 14000 nM T02728 CWI8C2 44447826 Ki = 47 nM T02728 C1KIX8 44447828 Ki = 210 nM T02728 CVH63S 44447863 Ki = 1.6 nM T02728 C3UE1C 44447864 Ki = 17 nM T02728 C34DVM 44447865 Ki = 30000 nM T02728 C4DL5C 44469677 IC50 > 10000 nM T02728 C94OME 44564776 EC50 = 2043 nM T02728 CATD40 44572613 Ki = 0.29 nM T02728 C0Y3CL 44572614 Ki = 0.73 nM T02728 CBG3K6 44572615 Ki = 4.87 nM T02728 CP63TW 44572616 EC50 = 1.85 nM T02728 CHM4V1 44572617 EC50 = 6.21 nM T02728 C6KWM1 44572618 EC50 = 57.7 nM T02728 CU0MQ4 44572619 EC50 = 7.96 nM T02728 C3TE2G 44572620 Ki = 4.5 nM T02728 CFI09D 44572621 EC50 = 6.44 nM T02728 C6RA9H 44572622 Ki = 2.99 nM T02728 CC2JK6 44572623 EC50 = 217 nM T02728 CSR9C1 44572624 Ki = 647 nM T02728 CZ96JA 44572625 Ki = 105 nM T02728 C9VA6D 44572626 EC50 = 1860 nM T02728 CW19UK 44572627 Ki = 631 nM T02728 CU47OK 44581036 IC50 = 3.76 nM T02728 CJ50IK 45102614 Ki = 28000 nM T02728 CQ7K3Y 45490651 EC50 = 6650 nM T02728 CM01RX 46890552 IC50 = 700 nM T02728 CN9KS4 46890553 IC50 = 8300 nM T02728 CF63HL 49798969 EC50 = 10.6 nM T02728 CMX46E 49837903 EC50 = 56000 nM T02728 C2S3KG 49837905 EC50 > 80000 nM T02728 C1LK8Y 49837907 EC50 > 80000 nM T02728 CX9M3E 49837912 EC50 = 298 nM T02728 C2P6TK 49837913 EC50 > 80000 nM T02728 CK2F0D 49837915 EC50 > 80000 nM T02728 CPB3C7 49837919 EC50 = 72000 nM T02728 CDW5G6 49837921 EC50 = 66000 nM T02728 CO61RX 49837922 EC50 > 80000 nM T02728 CA12GV 50898052 EC50 = 9200 nM T02728 C65CTG 50919363 EC50 = 5200 nM T02728 C7H2GT 50919365 EC50 = 3800 nM T02728 CICG82 50919370 EC50 = 46000 nM T02728 CD9J4Y 50919373 EC50 > 80000 nM T02728 C3RIF7 50919376 EC50 = 2300 nM T02728 CVQM43 51035368 EC50 = 12000 nM T02728 C65GEF 51035373 EC50 = 15000 nM T02728 C9YIZ5 52914819 EC50 = 12000 nM T02728 C6S9YI 52914822 EC50 = 18000 nM T02728 C3Y4DQ 52914826 EC50 > 80000 nM T02728 C9FJ6G 52951375 Ki = 47000 nM T02728 CL1E9Q 52951376 Ki = 2600 nM T02728 C2LOM8 52951377 Ki = 10000 nM T02728 CS3U7Z 52951476 Ki = 80000 nM T02728 C0XZ2V 52951477 Ki = 8300 nM T02728 CNI2F4 52951478 Ki = 32000 nM T02728 CC4U3O 53245521 EC50 = 10000 nM T02728 C3WTY4 53245542 EC50 = 30000 nM T02728 CE7A9B 53245571 EC50 = 5800 nM T02728 CH4EO6 53245574 EC50 = 34000 nM T02728 CMJ62D 53245590 EC50 = 2000 nM T02728 CQHV82 53245615 EC50 = 14000 nM T02728 C69HCK 53245626 EC50 = 23000 nM T02728 CB78FA 53495081 EC50 = 9400 nM T02728 CNFI86 54580106 Ki = 0.61 nM T02728 CPO5M6 54580107 Ki = 71 nM T02728 C6ZX1P 54580108 Ki = 1300 nM T02728 CYJ93A 54581089 Ki = 890 nM T02728 CP92RB 54582126 Ki = 0.23 nM T02728 CX7K3E 54582127 Ki = 3.4 nM T02728 CX90US 54583072 Ki = 26 nM T02728 CDXP96 54583073 Ki = 220 nM T02728 C2SCE8 54583074 Ki = 13000 nM T02728 CSN46R 54583075 Ki = 8.4 nM T02728 CCY5W1 54583076 Ki = 3700 nM T02728 CHSI63 54585021 Ki = 11 nM T02728 CHNT83 54585022 Ki = 1300 nM T02728 C24YLS 54585023 Ki = 8.4 nM T02728 C9I4DC 54585988 Ki = 4.6 nM T02728 CO0P4Z 54585989 Ki = 1100 nM T02728 CUQX42 54585990 Ki = 250 nM T02728 C0HI5E 54758538 EC50 = 17000 nM T02728 CZ63WS 54758539 EC50 = 8000 nM T02728 CC6F4U 56593272 EC50 = 20000 nM T02728 CY5VX7 56593273 EC50 = 7000 nM T02728 C1RJX8 56593274 EC50 > 80000 nM T02728 CX1N3I 56593278 EC50 = 4100 nM T02728 CMF4H8 56593279 EC50 = 68000 nM T02728 CB75SU 56593281 EC50 = 26000 nM T02728 C2J7VC 56593282 EC50 = 15000 nM T02728 CA9OV0 56593283 EC50 > 80000 nM T02728 C2FHP7 56593284 EC50 = 14000 nM T02728 CNG48L 56593288 EC50 = 35000 nM T02728 CY1N5C 56593289 EC50 = 45000 nM T02728 C7ZL2B 56593290 EC50 = 6100 nM T02728 CD06NY 56593291 EC50 = 25000 nM T02728 CQ60KY 56593292 EC50 > 80000 nM T02728 CNB83L 56593293 EC50 = 43000 nM T02728 C78BEX 56723766 EC50 = 9990 nM T02728 C3FB9E 71717277 Ki = 5.1 nM T02728 CWH6T3 72548703 IC50 = 0.25 nM T02728 CCG58A 72737612 Ki = 0.98 nM T02728 CD8F2O 73345472 IC50 = 59.6 nM T02728 CG62IS 73346308 EC50 > 80000 nM T02728 CU83RW 73346899 Ki = 3000 nM T02728 CO8S0I 73347807 EC50 > 80000 nM T02728 CH2YN5 73349346 EC50 = 17000 nM T02728 C6V7YB 73350917 EC50 = 23000 nM T02728 C8PZ4T 73352405 EC50 = 75000 nM T02728 C4G6FB 73353870 EC50 > 80000 nM T02728 C5IVA1 73355398 EC50 = 46000 nM T02728 CH02DL 73356134 IC50 = 0.4 nM T02728 CGTQ84 73356947 EC50 = 61000 nM T02728 CQ91AR 73356948 EC50 > 80000 nM T02728 C02BEM 76324673 EC50 = 970 nM T02728 CVTJ47 90236942 EC50 = 560 nM T02728 CV2ZA9 90237040 EC50 = 888 nM T02728 CYN71E 90237274 EC50 = 810 nM T02728 C32TFE 90237301 EC50 = 3360 nM T02728 C35UCB 90237332 EC50 = 732 nM T02728 C9XYG7 90237403 EC50 = 478 nM T02728 CJY78Q 90237466 EC50 = 710 nM T02728 CV5M9J 90237476 EC50 > 20000 nM T02728 C4EJG6 90237596 EC50 = 1040 nM T02728 C2IF0V 90237648 EC50 = 1120 nM T02728 C3H4ZK 90663196 IC50 = 0.5 nM T02728 C0V5EC 91826086 IC50 > 30000 nM T02728 CM12IY 101040509 Ki = 450 nM T02728 C2BZA6 101171051 IC50 = 15.2 nM T02728 CT0PR3 118610246 EC50 = 4230 nM T02728 CVTR06 118610255 EC50 = 3880 nM T02728 CV3WU8 118610260 EC50 = 810 nM T02728 CF1ZK7 118610278 EC50 = 10020 nM T02728 CU06NH 118610314 EC50 = 920 nM T02728 CMIO78 118610338 EC50 = 160 nM T02728 C2O7KY 118610372 EC50 = 1050 nM T02728 C4TI5F 118610386 EC50 = 2780 nM T02728 C5PI8K 118610402 EC50 = 500 nM T02728 CG9W0F 118610404 EC50 = 6720 nM T02728 CWB6J3 118610411 EC50 = 340 nM T02728 C07EYJ 118610423 EC50 = 270 nM T02728 CF29CD 118610426 EC50 = 160 nM T02728 CVHG45 118610427 EC50 = 1.18 nM T02728 CIC86N 118610470 EC50 = 1060 nM T02728 C23EKC 118617560 EC50 = 3010 nM T02728 C3YZP1 118617570 EC50 = 1720 nM T02728 CN64GY 118617599 EC50 = 590 nM T02728 C1M4LC 118617631 EC50 = 2230 nM T02728 CW81UC 118617645 EC50 = 560 nM T02728 CBH16N 118617715 EC50 = 1450 nM T02728 CY0QP8 118617724 EC50 = 1480 nM T02728 CYB18D 118617733 EC50 = 1260 nM T02728 CZ4EW5 118617765 EC50 = 990 nM T02728 CXWI39 118617781 EC50 = 1010 nM T02728 CA4U9L 118617787 EC50 = 440 nM T02728 CN75AR 118617789 EC50 = 640 nM T02728 CH1KM5 118617792 EC50 = 3810 nM T02728 C4OH7R 118617810 EC50 = 98 nM T02728 C9TR0S 118617901 EC50 = 600 nM T02728 CP2W0C 118617949 EC50 = 220 nM T02728 C89ZNS 118708030 EC50 = 2050 nM T02728 CZ62CD 118708031 EC50 = 25820 nM T02728 CP2O1Q 118708032 EC50 = 9440 nM T02728 CFM50J 118708033 EC50 = 15380 nM T02728 CSO50T 118708034 EC50 = 3260 nM T02728 CFI64D 118708035 EC50 = 9390 nM T02728 C3W1LJ 118708036 EC50 = 55070 nM T02728 CVE27J 118708037 EC50 = 4960 nM T02728 C36ZYC 118708038 EC50 = 3240 nM T02728 CTL0S5 118708039 EC50 = 7720 nM T02728 C5U1FS 118708040 EC50 = 24200 nM T02728 CV3YA5 118708041 EC50 = 2120 nM T02728 CV6U3W 118708042 EC50 > 100000 nM T02728 CK03NJ 118708043 EC50 > 100000 nM T02728 CP4H6G 118708044 EC50 = 5170 nM T02728 CKI4S5 118708045 EC50 > 100000 nM T02728 CWQ31H 118708046 EC50 > 100000 nM T02728 CMLE90 118708047 EC50 > 100000 nM T02728 C10VOG 118708048 EC50 = 4330 nM T02728 C0YP6K 118708049 EC50 > 100000 nM T02728 C5W4AS 118708050 EC50 > 100000 nM T02728 CDJ50Q 118708051 EC50 > 100000 nM T02728 C9TI5F 118708052 EC50 > 100000 nM T02728 C53ZNP 118708053 EC50 > 100000 nM T02728 CA2CU3 118708054 EC50 > 100000 nM T02728 CTA9F8 118708055 EC50 > 100000 nM T02728 CD7QY8 118708056 EC50 = 3280 nM T02728 C3Z4IG 118708057 EC50 = 2850 nM T02728 CA5X7R 118708058 EC50 = 7460 nM T02728 C9O6WP 122192055 EC50 = 26.6 nM T02728 C1DSL0 122192056 EC50 = 1.49 nM T02728 C3KWU5 122192057 EC50 = 0.34 nM T02728 C98IKC 122192058 IC50 = 968 nM T02728 C0A5VN 122192059 EC50 = 4.19 nM T02728 CFW0K8 122197318 IC50 = 3.4 nM T02728 C8Z2DE 122197319 IC50 = 0.6 nM T02728 C0LE9S 122197320 IC50 = 1.2 nM T02728 C2EW4P 127031263 Ki = 0.51 nM T02728 CO6T1L 127031275 Ki = 1.7 nM T02728 C2YNI4 127031283 Ki = 0.41 nM T02728 CEH29I 127031850 Ki = 0.36 nM T02728 CVZT87 127032101 Ki = 0.47 nM T02728 CCLG54 127032411 Ki = 0.47 nM T02728 CRS0K2 127033023 Ki = 0.26 nM T02728 CW4M5O 127033028 Ki = 0.59 nM T02728 C1GA4W 132547200 Ki = 20000 nM T02728 CW7V8Q 134134595 Ki = 35000 nM T02728 CIZ1T2 134136231 Ki = 67000 nM T02728 C07SHR 134138287 Ki = 53000 nM T02728 C8NFR1 134140868 Ki = 13000 nM T02728 CE5Z0K 134142369 Ki = 10000 nM T02728 C3S9GD 134143837 Ki = 72500 nM T02728 CK03XR 134144300 Ki = 5000 nM T02728 CMGT90 134145547 Ki = 870 nM T02728 C2KR6X 134145567 Ki = 10000 nM T02728 CHR4S3 134146201 Ki = 70500 nM T02728 CO8Q7F 134147225 Ki = 2170 nM T02728 CRH73L 134152554 Ki = 93 nM T02728 CKS0C3 134153118 Ki = 35000 nM T02728 C87ZMF 134155365 Ki = 7 nM T02728 C2MKS7 137645783 Ki > 10000 nM T02728 CY6N5R 137646112 Ki = 5700 nM T02728 COX29R 137651580 Ki > 10000 nM T02728 CN74UT 137651867 Ki = 455.6 nM T02728 CLF01S 137656771 Ki > 10000 nM T02728 CVP06T 137660279 Ki = 662.7 nM T02728 CPH2B4 145948619 Ki = 4.1 nM T02728 C3XDL0 145964771 EC50 = 182 nM T02728 C0CJP5 145966676 EC50 = 18 nM T02728 CMET14 145966776 EC50 = 166.2 nM T02728 C7IU2G 145967420 EC50 = 63 nM T02728 CZ5TN4 145970531 Ki > 10000 nM T02728 CU46LI 145970755 EC50 = 21 nM T02728 CA9MT7 145972052 EC50 = 24 nM T02728 CEI6M9 145974670 EC50 = 3 nM T02728 CRJ90L 145975472 Ki = 300 nM T02728 C3H5VJ 145975635 EC50 = 27 nM T02728 CGKX10 145976418 EC50 = 57 nM T02728 C7FVD0 145976898 EC50 = 7 nM T02728 CCM31K 145977513 EC50 = 15 nM T02728 C9JZ0U 145978385 Ki = 159 nM T02728 CB39KH 145979804 IC50 = 1700 nM T02728 CF64PV 145980057 IC50 = 1400 nM T02728 C74IAJ 145980071 IC50 = 14300 nM T02728 C6C7WK 145987656 IC50 > 100000 nM T02728 C0W4VP 145989581 IC50 = 17000 nM T02728 C8F0AP 145989745 EC50 = 166.3 nM T02728 CGF6C7 145989754 IC50 = 19800 nM T02728 C8PZ1Q 145990573 IC50 = 29800 nM T02728 CVIH91 145990648 IC50 = 10000 nM T02728 CY9F7A 145991532 IC50 = 7600 nM T02728 C0ITB3 145993831 IC50 > 100000 nM T02728 CA43NW 145994034 IC50 = 10300 nM T02728 COJ08U 155283653 EC50 = 6710 nM T02728 C6V2DS 155511768 Ki = 50 nM T02728 CA1Z7Y 155511940 Ki = 60 nM T02728 CXD67E 155513242 Ki = 9.333 nM T02728 C9FT0Y 155514775 Ki > 1000 nM T02728 CLUE10 155522776 Ki = 1.17 nM T02728 CAH73J 155525403 EC50 = 0.4169 nM T02728 CHZQ54 155529794 Ki = 0.7586 nM T02728 CYJT02 155543922 Ki = 3.548 nM T02728 CL7WT2 155544004 Ki = 0.28 nM T02728 CRVF36 155544464 Ki = 880 nM T02728 CRI8F0 155544586 IC50 = 63 nM T02728 CC6ZW3 155544972 Ki = 0.29 nM T02728 CY8XR1 155547077 Ki = 2.188 nM T02728 CLR03S 155547101 Ki = 9.333 nM T02728 CYX16L 155548706 EC50 = 0.3715 nM T02728 C02KMY 155548875 Ki = 4.074 nM T02728 CZOX60 155551503 Ki = 1.6 nM T02728 C9XU4F 155552814 Ki = 1 nM T02728 C2SA8V 155559775 EC50 = 1.023 nM T02728 C15GYE 155560503 Ki = 18 nM T02728 CE01TL 155560655 Ki = 0.88 nM T02728 C9U5VX 155561747 Ki = 2.512 nM T02728 CFTW36 155567371 IC50 = 60 nM T02728 CX25HK 155569027 Ki = 0.223 nM T02728 CY4IX3 155569268 Ki = 2.692 nM T02728 D00TPV 5311318 EC50 = 0.0416 nM T02728 D05ZUX 44207909 Ki >= 1000 nM T02728 D0B4SQ 44578945 Ki = 2.4 nM T02728 D0H7EB 44578944 Ki = 160 nM T02728 D0H8AI 25077406 IC50 = 0.2 nM T02728 D0N4RF 44413846 IC50 = 1.5 nM T02728 D0OJ7S 5311451 IC50 = 0.24 nM T02728 D0OT9G 44578943 Ki = 190 nM T02728 D0P5VL 11847007 IC50 = 0.14 nM T02728 D0S9PC 10102003 Ki = 0.51 nM T02728 D0T2RY 9948320 Ki >= 1000 nM T02728 D0V4HB 56661177 IC50 = 0.18 nM T02728 D0X3RW 44413847 IC50 = 0.51 nM T76286 C07XTF 52915134 IC50 = 0.2 ug.mL-1 T76286 CSAI17 52915252 IC50 = 1.5 ug.mL-1 T76286 C2NZ9F 52915254 IC50 = 2.4 ug.mL-1 T76286 CZC0L4 52915382 IC50 = 0.8 ug.mL-1 T76286 C5HXE6 52915498 IC50 = 2 ug.mL-1 T76286 CX1P3U 52916074 IC50 = 1.2 ug.mL-1 T73471 D05PHH 3447 IC50 = 383 nM T73471 D07XHO 4413 Ki = 0.53 nM T73471 D0M7JT 216210 Ki = 835 nM T73471 D0Y6SQ 2536 IC50 = 29 nM T73471 D04LWZ 761639 IC50 = 350 nM T73471 C2KE5Q 1508 Ki = 35000 nM T73471 CK9AZ0 122670 Ki = 500000 nM T73471 C6MQD0 124952 IC50 = 870 nM T73471 CZ17HE 445157 IC50 = 4460 nM T73471 CR4KE5 445844 IC50 = 2600 nM T73471 COK61H 639391 IC50 = 272 nM T73471 CN2B6S 6852211 Ki = 1580 nM T73471 CU8N3V 10578280 IC50 = 6550 nM T73471 C8NHR5 10984568 Ki = 3.38 nM T73471 CB1S5N 11363919 Ki = 553 nM T73471 CU07NO 11607091 Ki = 7400 nM T73471 CQ8OU1 13755335 IC50 = 3140 nM T73471 CMZ05T 44324727 Ki = 53100 nM T73471 CO46GL 44358382 IC50 > 10000 nM T73471 CC8S0D 44362303 IC50 = 6190 nM T73471 CE9I1R 44362422 Ki = 7000 nM T73471 CA90QH 91827690 Ki = 540 nM T73471 CZ0UR6 92220134 IC50 = 6490 nM T73471 C46MSP 118542774 Ki = 1120 nM T73471 C20WBY 118542785 Ki = 3400 nM T73471 CI65YK 118542879 Ki = 920 nM T73471 CEH93P 118542958 Ki = 690 nM T73471 CITU59 118548755 Ki = 1100 nM T73471 CMF5R6 118548758 Ki = 210 nM T73471 C1IH2W 118548759 Ki = 760 nM T73471 C6LZQ3 118548760 Ki = 720 nM T73471 C62ZNW 118548761 Ki = 670 nM T73471 C3WQ9D 118548776 Ki = 310 nM T73471 CU01RP 118548813 Ki = 530 nM T73471 C7NG3I 118721642 Ki = 0.22 nM T73471 CTV97I 118721643 Ki = 0.41 nM T73471 C1NS7F 118721644 Ki = 0.21 nM T73471 C3OCD1 118721645 Ki = 0.58 nM T73471 CQK2U8 118721646 Ki = 2.1 nM T73471 C4HB3G 118721647 Ki = 0.28 nM T73471 CNP30X 118721648 Ki = 0.34 nM T73471 CRPV34 118721649 Ki = 0.57 nM T73471 CU5KB2 118721650 Ki = 0.21 nM T73471 CJA76N 118721651 Ki = 1.2 nM T73471 CS3GX9 118721652 Ki = 0.6 nM T73471 C0Y9EU 118721653 Ki = 0.55 nM T73471 CJ4FI3 118721654 Ki = 8.5 nM T73471 CK2QX9 118721655 Ki = 1.4 nM T73471 C4UYE3 118721656 Ki = 0.68 nM T73471 CP9L7H 118721657 Ki = 0.61 nM T73471 C2MI1J 118721658 Ki = 1.2 nM T73471 CIPY54 118721659 Ki = 0.47 nM T73471 CSAZ58 118728084 Ki = 1200 nM T73471 C4K6HY 118729129 Ki = 3500 nM T73471 C4MX0T 118729130 Ki = 2600 nM T73471 CUC7N1 118729131 Ki = 2400 nM T73471 C1KWF0 118729132 Ki = 7400 nM T73471 CS7QD3 118729855 Ki = 3300 nM T73471 CWK9I0 118729856 Ki = 1000 nM T73471 C73DSK 118729857 Ki = 2300 nM T73471 CM2E0V 118729858 Ki = 48 nM T73471 C63TEA 118729859 Ki = 4700 nM T73471 CPD68M 118729860 Ki = 670 nM T73471 C3NK4O 121232387 Ki = 100 nM T73471 CG4LR5 122194707 Ki = 4900 nM T73471 CA6U5Q 122194708 Ki = 4800 nM T73471 CZ8CH4 122194709 Ki = 1400 nM T73471 CLDC14 122194710 Ki = 600 nM T73471 C6NGM7 122194711 Ki = 400 nM T73471 CR4CY8 122194712 Ki = 100 nM T73471 COY83A 122535266 Ki = 831 nM T73471 CG5S2R 122535267 Ki = 116 nM T73471 CAI69W 123238067 Ki = 760 nM T73471 C76BAD 123424620 Ki = 560 nM T73471 CDN27U 124557571 IC50 > 10000 nM T73471 CA30BN 127033248 Ki = 61200 nM T73471 CO7PY0 127033521 Ki = 15100 nM T73471 CE0QZ4 127033522 Ki = 20800 nM T73471 C7ZIR9 127034099 Ki = 2120 nM T73471 CUW45R 127037924 Ki > 10000 nM T73471 CG13JW 127037925 Ki > 10000 nM T73471 C5HV9L 127037926 Ki > 10000 nM T73471 CTJP37 127042186 Ki = 0.83 nM T73471 C8AS4D 127042541 Ki = 1.04 nM T73471 CVN74W 127042542 Ki = 2.88 nM T73471 CP5AG8 127042543 Ki = 22.4 nM T73471 CW8ML6 127042544 Ki = 21.5 nM T73471 C3SRT7 127042545 Ki > 10000 nM T73471 CC24ST 127042546 Ki = 2.91 nM T73471 CQ9OB0 127044670 IC50 = 23000 nM T73471 COS19G 127044671 IC50 = 5900 nM T73471 C9E6KQ 127044672 IC50 = 11000 nM T73471 C4FRL2 127044841 IC50 = 9300 nM T73471 CK28IC 127044842 IC50 = 8900 nM T73471 C9XZR3 127044843 IC50 = 7300 nM T73471 CFL17D 127044844 IC50 = 14000 nM T73471 CS21GF 127045102 IC50 = 70000 nM T73471 CWO5G1 134130685 IC50 = 2800 nM T73471 CD06PE 134313025 Ki = 0.16 nM T73471 CRE5O9 145960395 IC50 = 58000 nM T73471 C0M2QA 145960406 IC50 = 3000 nM T73471 CRK0L6 145960477 IC50 = 90 nM T73471 C0OF9H 145960548 IC50 = 5000 nM T73471 C84PHM 145960637 IC50 = 220 nM T73471 C36PYJ 145960730 IC50 = 1100 nM T73471 CW9X7P 145960760 IC50 = 22 nM T73471 C47IGD 145960856 IC50 = 860 nM T73471 CXI16W 145960913 IC50 = 250 nM T73471 C41LXH 145960914 IC50 = 330 nM T73471 C02KUI 145961020 IC50 = 300 nM T73471 CK7H3W 145961084 IC50 = 3150 nM T73471 CYS02N 145961266 IC50 = 4020 nM T73471 C25NZG 145961305 IC50 = 900 nM T73471 CG6R0N 145961689 IC50 = 100 nM T73471 CXUW40 145961875 IC50 > 19000 nM T73471 CD0I6N 145962360 IC50 = 11000 nM T73471 CGV68W 145962449 IC50 = 600 nM T73471 COXY65 145962472 IC50 = 38 nM T73471 C39NWG 145962609 IC50 = 2000 nM T73471 CZN4A5 145962690 IC50 = 1400 nM T73471 CJ6Y4W 145962813 IC50 = 500 nM T73471 CR78WU 145963185 IC50 = 73000 nM T73471 C93BRK 145963190 IC50 = 1500 nM T73471 CD31BO 145963222 IC50 = 700 nM T73471 CA8J7F 145963231 IC50 = 1800 nM T73471 CJP64T 155510867 IC50 = 5 nM T73471 CUP78D 155512098 IC50 = 20 nM T73471 C1RYT8 155517297 Ki = 228 nM T73471 CX6C5Y 155520312 IC50 = 60 nM T73471 CE01NY 155523107 IC50 = 10 nM T73471 CW9K3R 155523263 IC50 = 8 nM T73471 CGMP07 155523803 Ki = 0.09 nM T73471 C4HN6V 155525157 Ki = 180 nM T73471 C7SB9X 155528083 Ki = 256 nM T73471 CG68UH 155529134 IC50 = 20 nM T73471 CN0B2S 155529433 Ki = 1.7 nM T73471 C5QT3D 155529505 Ki = 98 nM T73471 CA82SM 155530516 Ki = 0.67 nM T73471 CER1Z8 155532768 Ki = 372 nM T73471 C1HAW5 155533558 IC50 = 2 nM T73471 CEFK81 155534191 Ki = 104 nM T73471 C7M2UT 155534310 IC50 = 0.6 nM T73471 C2YB0P 155535378 Ki = 555 nM T73471 C6AE0I 155535379 Ki = 125 nM T73471 CUV1I4 155535874 IC50 = 110 nM T73471 CT4S3M 155544624 IC50 = 90 nM T73471 C5FZ3I 155545003 Ki = 302 nM T73471 CA08GE 155545013 Ki = 764 nM T73471 CQ51DI 155546002 IC50 = 0.5 nM T73471 CK0E7M 155548720 IC50 = 70 nM T73471 C3R9TO 155551160 IC50 = 60 nM T73471 CM3X6Y 155555703 Ki = 226 nM T73471 CXYR84 155556203 Ki = 227 nM T73471 CM63SG 155557605 IC50 = 70 nM T73471 C0IW5Z 155557962 IC50 = 110 nM T73471 C3VJ5W 155559076 Ki = 240 nM T73471 CY60RV 155559158 Ki = 67 nM T73471 CQ3MJ4 155559840 Ki = 102 nM T73471 C0B3ID 155562970 Ki = 391 nM T73471 CTF0S7 155566456 Ki = 0.27 nM T73471 D06MTX 1506 Ki = 40000 nM T73471 D08KCA 72429 Ki = 61 nM T73471 D0W2SV 70689167 Ki = 1.1 nM T92144 D01PZD 5329098 IC50 > 10000 nM T92144 D03ZBT 11626560 IC50 = 5 nM T92144 D09GDD 11167602 IC50 = 1.5 nM T92144 D0G6QF 3081361 IC50 = 567 nM T92144 D0IQ6P 25102847 IC50 = 14.3 nM T92144 D0J9ZR 4477 IC50 = 67800 nM T92144 D0OB0F 5328940 IC50 = 1191 nM T92144 D0W5HK 216239 IC50 = 0.39 nM T92144 D00YPR 9811611 IC50 = 18 nM T92144 D02UFQ 11620908 IC50 > 10000 nM T92144 D03LWG 53235510 IC50 = 2051 nM T92144 D0D1GF 42642645 IC50 = 1.1 nM T92144 D0E3TC 44259 IC50 = 50.9 nM T92144 D0FA6S 54576299 IC50 = 8 nM T92144 D0FD6D 11751922 IC50 = 50 nM T92144 D0IQ0Z 46885626 IC50 = 59 nM T92144 D0M9QZ 11485656 IC50 = 170 nM T92144 D0O6WV 24794418 IC50 > 500 nM T92144 D0YK9D 9956119 IC50 > 5000 nM T92144 D09HEV 6539952 IC50 = 250 nM T92144 D0F8DL 176155 IC50 = 20000 nM T92144 D0H4GI 10275001 IC50 > 10000 nM T92144 D0L5YF 5329032 IC50 > 100000 nM T92144 D0T3ME 156422 IC50 = 25 nM T92144 CB1VW3 1400 IC50 = 7000 nM T92144 C63WLY 89644 IC50 = 8.9 ug.mL-1 T92144 C5JE2Z 104860 IC50 = 8.8 ug.mL-1 T92144 C6Y9CV 151193 IC50 > 10000 nM T92144 CI1NA5 159926 IC50 = 1.9 ug.mL-1 T92144 CYBA43 177458 IC50 = 4.5 ug.mL-1 T92144 CP71KC 683649 IC50 > 10000 nM T92144 CDSN72 838889 IC50 = 1000 nM T92144 CCN9D5 3142817 IC50 = 3000 nM T92144 C0RXL8 5326956 IC50 = 1.995 nM T92144 CFW19M 5329009 IC50 = 8300 nM T92144 CYUA16 5329801 IC50 > 20000 nM T92144 C19VND 5329802 IC50 > 20000 nM T92144 CI6BY0 5329803 IC50 = 1780 nM T92144 CD0V3Y 5329804 IC50 = 540 nM T92144 CO7SF0 5329805 IC50 = 1480 nM T92144 C98ZEL 5329806 IC50 = 300 nM T92144 CB1DR2 5329807 IC50 = 600 nM T92144 CXS32G 5329808 IC50 = 190 nM T92144 C6NFY4 5329809 IC50 > 20000 nM T92144 CKOJ45 5329810 IC50 = 501 nM T92144 C8TEO1 5329811 IC50 = 851.14 nM T92144 C17MYA 5329812 IC50 = 28 nM T92144 CPBG38 5329813 IC50 = 21.88 nM T92144 CZTJ18 5329814 IC50 = 58.88 nM T92144 C5CY9J 5329815 IC50 = 275 nM T92144 C5RK3H 5330188 IC50 = 17100 nM T92144 CD7U5B 5330196 IC50 = 11300 nM T92144 CB23PA 5330197 IC50 = 11300 nM T92144 CDQ3M7 5359485 IC50 = 7 ug.mL-1 T92144 C54BYP 5360741 IC50 = 3.5 ug.mL-1 T92144 C2DCW3 5916724 IC50 = 6000 nM T92144 CB7WK3 5938113 IC50 = 1800 nM T92144 CA31PJ 6539953 IC50 = 750 nM T92144 C64ZJA 6539954 IC50 = 606 nM T92144 CBD1H7 6539955 IC50 = 5730 nM T92144 CWHY29 6539956 IC50 = 4680 nM T92144 CW76RA 6539957 IC50 = 521 nM T92144 C7K1QS 6539958 IC50 = 933 nM T92144 CJ7IL2 6539959 IC50 = 137 nM T92144 CAE95J 6539960 IC50 = 888 nM T92144 CH86XJ 6539961 IC50 = 1130 nM T92144 C41FUH 6539962 IC50 = 2450 nM T92144 C7M2JP 6539963 IC50 = 1440 nM T92144 CS5V1C 6539964 IC50 = 910 nM T92144 C10FYS 6539966 IC50 = 1020 nM T92144 CIS1T3 6539967 IC50 = 203 nM T92144 CTZ4W0 6539971 IC50 = 1200 nM T92144 CAOU70 6539972 IC50 = 110 nM T92144 CE9L8Y 6539983 IC50 = 338.84 nM T92144 CUPQ08 6539985 IC50 = 720 nM T92144 CK9TD3 6539988 IC50 = 1288.25 nM T92144 CDA25S 6539989 IC50 = 891.25 nM T92144 C6Q4ZY 6539990 IC50 = 912.01 nM T92144 C3SXL8 6539991 IC50 = 360 nM T92144 CWC68D 6539992 IC50 = 1584.89 nM T92144 CR9GL1 6539993 IC50 = 1000 nM T92144 CK23SV 6539994 IC50 = 398.11 nM T92144 C9ZN6H 6539995 IC50 = 850 nM T92144 C39QGE 6539996 IC50 = 891.25 nM T92144 C8EJI1 6539997 IC50 = 210 nM T92144 CYQ9D4 6539998 IC50 = 1200 nM T92144 CH2EV5 6539999 IC50 = 128.82 nM T92144 C9GMT4 6540000 IC50 = 1096.48 nM T92144 CWA5M6 6540001 IC50 = 100 nM T92144 C3SAD6 6540002 IC50 = 512.86 nM T92144 CU14NK 6540003 IC50 = 169.82 nM T92144 CIC64F 6540004 IC50 = 360 nM T92144 CMEZ23 6540005 IC50 = 16.98 nM T92144 CG1L6R 6540006 IC50 = 120 nM T92144 C92OFS 6540007 IC50 = 467.74 nM T92144 C7H4QP 6540008 IC50 = 140 nM T92144 CF97JX 6540009 IC50 = 426.58 nM T92144 C52OIP 6540010 IC50 = 630 nM T92144 C2O4MX 6540012 IC50 = 288.4 nM T92144 C6HWM9 6540013 IC50 = 575.44 nM T92144 CB9N7T 6540014 IC50 = 870.96 nM T92144 CSGQ06 6540015 IC50 = 250 nM T92144 CP32OT 6540016 IC50 = 270 nM T92144 C4NWO7 6540017 IC50 = 257.04 nM T92144 C8AU3M 6540018 IC50 = 218.78 nM T92144 C3K7TM 6540019 IC50 = 110 nM T92144 CM1TH0 6540020 IC50 = 190 nM T92144 CP0XI6 6603792 IC50 = 1980 nM T92144 CSM34J 9804627 IC50 = 12160 nM T92144 C41QWA 9857146 IC50 > 10000 nM T92144 CQ64LI 9935852 IC50 = 10 nM T92144 CP2S5A 9936664 IC50 = 1357 nM T92144 CS5KX9 9938299 IC50 = 17 nM T92144 C54ZXH 9950678 IC50 = 2680 nM T92144 C5LA8Y 9958299 IC50 = 6.3 nM T92144 CUJR40 10062694 EC50 = 200 nM T92144 C7TA9J 10113568 IC50 = 18.3 nM T92144 CV67EI 10117977 IC50 = 1.5 nM T92144 CT96JK 10120050 IC50 = 16 nM T92144 C3JGH7 10141033 IC50 = 2.6 nM T92144 CNRX37 10142514 IC50 = 11 nM T92144 C3FGO2 10160775 IC50 = 18 nM T92144 CIQG50 10161259 IC50 = 71 nM T92144 C5QHB6 10161543 IC50 = 21380 nM T92144 C3TZ1Y 10163749 IC50 = 8 nM T92144 C29JTQ 10164190 IC50 = 6.5 nM T92144 C1Q6OJ 10166498 IC50 = 2.8 nM T92144 CC78NE 10179293 IC50 = 746 nM T92144 C7GN8Q 10183216 IC50 = 56 nM T92144 CU0WT6 10184615 IC50 = 2.6 nM T92144 CJU67H 10186182 IC50 = 41 nM T92144 CZI8M7 10186183 IC50 = 5600 nM T92144 C1KNM3 10186269 IC50 = 10 nM T92144 CCXY21 10204357 IC50 = 40 nM T92144 CYW95D 10206527 IC50 = 6.4 nM T92144 C1VUP6 10229632 IC50 = 41 nM T92144 CZX26W 10230568 IC50 = 5.2 nM T92144 CF90MC 10230609 IC50 = 3200 nM T92144 C1A5HT 10233129 IC50 = 85 nM T92144 CC9E5Q 10249989 IC50 = 700 nM T92144 C2F6DJ 10275349 IC50 = 60 nM T92144 CJGH26 10275985 IC50 = 4130 nM T92144 C5HC0D 10276395 IC50 > 10000 nM T92144 C12YUR 10278843 IC50 = 20 nM T92144 C60ZOC 10278844 IC50 = 91 nM T92144 CTHI58 10279624 IC50 = 6.5 nM T92144 C10UBJ 10280848 IC50 = 160 nM T92144 CFY14M 10300768 IC50 = 28 nM T92144 CP1LO7 10302209 IC50 = 60 nM T92144 C4J9ON 10309830 IC50 = 300 nM T92144 CY7WK8 10314049 IC50 = 3000 nM T92144 C9ZXG2 10357919 IC50 = 2700 nM T92144 CS1H7L 10362983 IC50 = 540 nM T92144 C4CV5L 10470475 IC50 = 1800 nM T92144 C8TA4Z 11129889 IC50 = 14000 nM T92144 CX0QO7 11192412 IC50 = 15 nM T92144 C8T2NG 11211389 IC50 = 5300 nM T92144 CT3K9Z 11213588 IC50 = 1 nM T92144 C5F2PA 11213751 IC50 = 58 nM T92144 CG29JX 11214363 IC50 = 43 nM T92144 CQ4XT3 11224593 IC50 = 8300 nM T92144 CVOW82 11238420 IC50 = 10100 nM T92144 CZS41D 11260323 IC50 = 241 nM T92144 C6C3JX 11281930 IC50 > 20000 nM T92144 C2IA4K 11294266 IC50 = 43 nM T92144 CGP80V 11328586 IC50 = 386 nM T92144 CEC31B 11351900 IC50 = 1000 nM T92144 CQ6M1W 11352718 IC50 = 568 nM T92144 CB45PJ 11362483 IC50 = 25000 nM T92144 C9B4XP 11363872 IC50 = 9 nM T92144 C25ZCN 11374110 IC50 = 270 nM T92144 CJ75ZF 11375010 IC50 = 72 nM T92144 CP4ZO0 11375301 IC50 = 110 nM T92144 C4IH5E 11383525 IC50 = 8300 nM T92144 CT3VP7 11398307 IC50 = 121 nM T92144 CEV1O4 11398610 IC50 = 2188 nM T92144 C8TIS2 11420237 IC50 = 24 nM T92144 C73PUW 11420344 IC50 = 260 nM T92144 CREQ51 11429654 IC50 = 249 nM T92144 CY0A4E 11429729 IC50 = 1000 nM T92144 CFJ6B2 11441375 IC50 = 25000 nM T92144 C1LU5O 11443317 IC50 = 20 nM T92144 C2ZO1F 11443318 IC50 = 63 nM T92144 CT2L6G 11443940 IC50 = 13 nM T92144 CL2BZ5 11454462 IC50 = 26 nM T92144 C4Q7XD 11474276 IC50 = 25000 nM T92144 C4NR2I 11476141 IC50 = 136 nM T92144 C2Z7WP 11486459 IC50 = 25000 nM T92144 C80QYI 11497471 IC50 = 1 nM T92144 C8AY3B 11518031 IC50 = 3.6 nM T92144 CO70EZ 11526166 IC50 = 13 nM T92144 CL7X4Q 11530963 IC50 = 2800 nM T92144 CN1K3R 11545702 IC50 = 3 nM T92144 CACS26 11561968 Ki > 2000 nM T92144 CA2KX0 11590078 IC50 = 8100 nM T92144 CONZ37 11591872 IC50 = 33 nM T92144 C69FYK 11604142 Ki = 200 nM T92144 CY6SW0 11617856 IC50 = 1220 nM T92144 CUO43M 11620207 IC50 = 21 nM T92144 C5B3XJ 11620410 IC50 = 3180 nM T92144 C70LDZ 11625929 IC50 = 2 nM T92144 C9ZD2E 11626406 IC50 > 8333 nM T92144 CWM80X 11627419 IC50 = 13 nM T92144 CVH29N 11642023 IC50 = 220 nM T92144 CTNK57 11648060 IC50 = 504 nM T92144 CRV5D2 11655925 IC50 = 43 nM T92144 CQ47BI 11662314 IC50 = 510 nM T92144 CCGO58 11669282 IC50 = 623 nM T92144 CPME86 11670863 IC50 = 37 nM T92144 CW9B8E 11678175 IC50 = 181 nM T92144 CJ9KN7 11683817 IC50 > 10000 nM T92144 CP3U0W 11684933 IC50 > 25000 nM T92144 CYO6X9 11684994 Ki = 200 nM T92144 CCEY64 11689855 IC50 = 47 nM T92144 CU0E8O 11690457 Ki > 2000 nM T92144 CB0AP2 11705863 Ki > 2000 nM T92144 C9ROB0 11713267 IC50 = 8 nM T92144 CZY05V 11719421 IC50 = 678 nM T92144 CL7B9U 11724621 IC50 = 13000 nM T92144 CRZ4K6 11724734 IC50 = 55000 nM T92144 CK97YQ 11744026 IC50 = 1400 nM T92144 CS5QL4 11749561 IC50 = 25000 nM T92144 CV64JS 11750694 IC50 = 1800 nM T92144 CE0KI4 11753519 IC50 = 570 nM T92144 CP7AH3 11755812 IC50 = 67 nM T92144 C63GPF 11775935 IC50 = 18000 nM T92144 CS36BH 11843159 IC50 = 200 nM T92144 CHR92S 11858109 IC50 = 26 nM T92144 CM50UH 12000646 EC50 = 540 nM T92144 CU4C3V 12968172 IC50 = 23400 nM T92144 CI8VE5 12968173 IC50 = 11100 nM T92144 CR75GZ 12968174 IC50 = 1810 nM T92144 CEVY69 12968175 IC50 = 500 nM T92144 CL1PR6 12968176 IC50 = 360 nM T92144 CY5EA7 12968177 IC50 = 610 nM T92144 CZ98FV 12968178 IC50 = 2260 nM T92144 C4SUK6 12968179 IC50 = 130 nM T92144 CGIZ84 12968180 IC50 = 410 nM T92144 C5MX8N 12968181 IC50 = 580 nM T92144 CDGF78 15282555 IC50 = 800 nM T92144 C7LB4I 15949613 IC50 = 20 nM T92144 C9RQN8 15950748 IC50 > 25000 nM T92144 CSK90Y 15991573 IC50 = 1 nM T92144 C8PRQ6 16040281 IC50 = 17 nM T92144 CFWR47 16040288 IC50 = 68 nM T92144 C7NCA6 16040289 IC50 >= 25000 nM T92144 C4MQU1 16040290 IC50 = 10 nM T92144 CQI0A5 16043229 IC50 = 259 nM T92144 CZKD04 16043241 IC50 = 415 nM T92144 C9X4TQ 16043242 IC50 = 19 nM T92144 C9TU1O 16046126 IC50 > 1000 nM T92144 CI74HE 16049888 IC50 = 11 nM T92144 CVE6C8 16086088 IC50 = 1.8 nM T92144 C73MLJ 16108977 IC50 < 1 nM T92144 C01GIO 16108981 IC50 = 22 nM T92144 C6FO0H 16108986 IC50 = 153 nM T92144 CXI9C8 16108987 IC50 = 2700 nM T92144 CEC7P3 16108988 IC50 = 103 nM T92144 CGK5O8 16108989 IC50 = 366 nM T92144 C5SE6X 16108990 IC50 = 399 nM T92144 C03GLR 16108991 IC50 = 4 nM T92144 C3L6TH 16108992 IC50 = 111 nM T92144 COEI61 16108993 IC50 > 25000 nM T92144 C39YWL 16108994 IC50 > 25000 nM T92144 C9IX0U 16108995 IC50 = 39 nM T92144 CU2TK3 16108996 IC50 = 40 nM T92144 CA2U9H 16108997 IC50 = 4 nM T92144 CX21ZN 16108999 IC50 = 140 nM T92144 CF57NZ 16109000 IC50 = 53 nM T92144 CQG45C 16109001 IC50 = 30 nM T92144 C3L8KE 16109002 IC50 = 6 nM T92144 CM40ZW 16109003 IC50 = 13 nM T92144 C8P4ZK 16109016 IC50 = 11 nM T92144 CY1E3Q 16109017 IC50 = 39 nM T92144 CV7S6Z 16109018 IC50 = 17 nM T92144 CB98HV 16109019 IC50 = 44 nM T92144 C49VTS 16109020 IC50 = 14 nM T92144 C6FZ7A 16109023 IC50 = 3 nM T92144 CWS8D0 16109024 IC50 = 85 nM T92144 C1WS6E 16109034 IC50 = 250 nM T92144 C8IES6 16109035 IC50 = 620 nM T92144 C1U8XW 16109036 IC50 = 8 nM T92144 CNG5L6 16109037 IC50 = 140 nM T92144 C34KRB 16109040 IC50 = 10 nM T92144 CZ5Y3V 16116847 IC50 > 25000 nM T92144 CLO43V 16116849 IC50 > 25000 nM T92144 C0HO6T 16118191 IC50 > 8300 nM T92144 CT92BZ 16118192 IC50 > 8300 nM T92144 CIZ6B4 16118193 IC50 = 6078 nM T92144 C2CN5O 16118323 IC50 > 8300 nM T92144 C4GTU3 16118324 IC50 > 8300 nM T92144 CXC78K 16118603 IC50 > 25000 nM T92144 CI4E6Y 16118605 IC50 > 25000 nM T92144 C8LIW4 16118609 IC50 > 25000 nM T92144 CGC34R 16118737 IC50 = 9950 nM T92144 CAN2K6 16118739 IC50 > 25000 nM T92144 CZ08YH 16214904 IC50 = 47 nM T92144 CP3HS4 16220354 IC50 = 4600 nM T92144 CU56EW 16664858 IC50 > 10000 nM T92144 C0VUQ3 16727122 IC50 = 1357 nM T92144 C6S3YO 16731782 IC50 = 27 nM T92144 CK9CV4 16733534 IC50 = 2 nM T92144 CDZ31W 16747696 IC50 = 4877 nM T92144 CL9BQ6 17748275 IC50 = 33 nM T92144 CI10AY 17755137 IC50 = 3200 nM T92144 C4HLX0 17755232 IC50 = 13 nM T92144 CU9MH8 17755233 IC50 = 130 nM T92144 C04GML 17755327 IC50 = 3200 nM T92144 CIS52L 17755330 IC50 = 71 nM T92144 CQ5D9H 17755420 IC50 = 3.7 nM T92144 CQ19GV 17755641 IC50 = 2190 nM T92144 CL39DG 17755642 IC50 = 680 nM T92144 C1JFM0 17755746 IC50 = 5400 nM T92144 C1L5IA 17755861 IC50 = 4.9 nM T92144 C0WEF9 17965846 IC50 = 1400 nM T92144 CJA0D6 18451024 IC50 = 3700 nM T92144 C6FQB7 18451036 IC50 > 50000 nM T92144 C5WAV7 19597382 IC50 = 600 nM T92144 CU5CK6 19597400 IC50 = 3400 nM T92144 CZQ92B 19597433 IC50 = 430 nM T92144 C02JLX 19597448 IC50 = 900 nM T92144 CYIX85 19597450 IC50 = 560 nM T92144 CFH4I2 19597457 IC50 = 1900 nM T92144 CIBE65 19597460 IC50 = 16710 nM T92144 C0JQ7H 19597465 IC50 = 1220 nM T92144 CP01WN 19597468 IC50 = 600 nM T92144 CA09JB 19597476 IC50 = 400 nM T92144 CC78WA 19597518 IC50 = 4900 nM T92144 CV0U1N 19597532 IC50 = 1500 nM T92144 C1B3DX 19597536 IC50 = 1800 nM T92144 CV7C2K 20817018 IC50 = 1020 nM T92144 CQ5X7V 20817081 IC50 = 520 nM T92144 CLOR96 22736225 IC50 = 6620 nM T92144 CT39NL 22736235 IC50 = 58.3 nM T92144 CAU62I 22736238 IC50 > 50000 nM T92144 CV1OI5 22736332 IC50 = 5150 nM T92144 C5ONK2 22736361 IC50 = 11620 nM T92144 C9QLP0 23133323 IC50 = 2500 nM T92144 CJ5N1R 23625762 IC50 = 250 nM T92144 C96KQX 23646931 IC50 = 99 nM T92144 C6UJ1B 23646932 IC50 = 62 nM T92144 C2MJ3D 23646933 IC50 = 30 nM T92144 C8YL1K 23646935 IC50 = 10 nM T92144 CSFK63 23646936 IC50 = 380.19 nM T92144 CEN96M 23646937 IC50 = 407.38 nM T92144 CJ5H1Z 23646938 IC50 = 10.23 nM T92144 CIP7T2 23646939 IC50 = 204.17 nM T92144 CL4ST0 23646940 IC50 = 223.87 nM T92144 C4E2OX 23646941 IC50 = 181.97 nM T92144 CI32JB 23646942 IC50 = 81.28 nM T92144 CI6C1R 23658582 IC50 > 5000 nM T92144 C2RV3U 24180608 IC50 = 12 nM T92144 CHU49V 24757938 IC50 = 580 nM T92144 C7YG1N 24759534 IC50 = 4700 nM T92144 CAJ4T2 24762205 IC50 = 1000 nM T92144 CQNP54 24764449 IC50 = 1000 nM T92144 CCPS81 24764502 IC50 > 35000 nM T92144 C4Z9CN 24769780 IC50 = 221 nM T92144 CO9Z0H 24822598 IC50 = 9400 nM T92144 C51IZL 24822599 IC50 = 1400 nM T92144 CA90EF 24822600 IC50 = 25000 nM T92144 C4A6LB 24823090 IC50 = 1100 nM T92144 C2B4JP 24823091 IC50 = 25000 nM T92144 CF6M3W 24823093 IC50 = 7400 nM T92144 C0NLO8 24823094 IC50 = 8300 nM T92144 C7D8PC 24823095 IC50 = 25000 nM T92144 C14FLQ 24823250 IC50 = 25000 nM T92144 C3KPO7 24823251 IC50 = 8300 nM T92144 C36BFD 24823252 IC50 = 8300 nM T92144 CBF60S 24823253 IC50 = 25000 nM T92144 CYBI02 24823426 IC50 > 5000 nM T92144 C45UGH 24823586 IC50 = 123 nM T92144 CFA3T8 24823588 IC50 > 25000 nM T92144 C51ZTV 24823589 IC50 > 25000 nM T92144 CX0QC1 24823590 IC50 > 8300 nM T92144 CR7CH6 24823736 IC50 > 25000 nM T92144 C26KXV 24823738 IC50 > 25000 nM T92144 CO3K7R 24823740 IC50 > 5000 nM T92144 CBLJ48 24823898 IC50 > 25000 nM T92144 CG0K1Z 24824046 IC50 > 25000 nM T92144 CDT3L2 24824050 IC50 = 1600 nM T92144 CLN48F 24824051 IC50 = 1500 nM T92144 C0NXE2 24824052 IC50 > 4000 nM T92144 CWTI12 24824188 IC50 > 4000 nM T92144 CQ1A8W 24824189 IC50 = 430 nM T92144 C8RE5C 24824190 IC50 > 4000 nM T92144 C3K1FM 24824191 IC50 > 4000 nM T92144 CV0S5L 24824318 IC50 = 2200 nM T92144 CUK14T 24824319 IC50 > 4000 nM T92144 CZ09ID 24824320 IC50 > 4000 nM T92144 CM28KX 24824321 IC50 > 4000 nM T92144 CD57UN 24824322 IC50 = 1500 nM T92144 CNI50G 24824323 IC50 > 4000 nM T92144 C84VZK 24824448 IC50 = 4000 nM T92144 C6OC4K 24824449 IC50 = 4300 nM T92144 C5BA7V 24824452 IC50 = 290 nM T92144 CR49SP 24824453 IC50 > 4000 nM T92144 CG64EL 24824454 IC50 > 4000 nM T92144 CCS58O 24863072 IC50 = 200 nM T92144 C6C2GX 24863500 IC50 = 5.8 nM T92144 CYVB83 24863584 IC50 = 8.1 nM T92144 CQ15ML 24863670 IC50 > 1000 nM T92144 C4XZ3N 24863671 IC50 > 1000 nM T92144 C4MG3B 24882476 IC50 = 3440 nM T92144 CFK2B9 24882503 IC50 = 300 nM T92144 C43HWQ 24883287 IC50 = 5000 nM T92144 C8DA5Q 24883334 IC50 = 2200 nM T92144 C4V9GH 24894117 IC50 = 5200 nM T92144 CHVU39 24894885 IC50 = 48000 nM T92144 CZ6KD4 24894886 IC50 = 26000 nM T92144 CKBY19 24894887 IC50 = 25000 nM T92144 C57BHF 24894888 IC50 = 24000 nM T92144 CB5TP8 24894992 IC50 = 11000 nM T92144 C32SUJ 24894993 IC50 = 11000 nM T92144 C38TGD 24894994 IC50 = 31000 nM T92144 CP7QT2 24894995 IC50 = 34000 nM T92144 C41SIT 24894996 IC50 = 11000 nM T92144 CFW40U 24894997 IC50 = 1700 nM T92144 CF4N9X 24895100 IC50 = 25000 nM T92144 CN13JF 24899915 IC50 = 6.8 ug.mL-1 T92144 CBWR97 24899916 IC50 = 1.4 ug.mL-1 T92144 C9F2JD 24899917 IC50 > 10 ug.mL-1 T92144 C64MTI 24900160 IC50 = 3.8 ug.mL-1 T92144 CO2I6Q 24900161 IC50 > 10 ug.mL-1 T92144 CT8OF0 24983254 IC50 = 16 nM T92144 CVF62Q 24983255 IC50 = 44 nM T92144 CX6FR3 24983298 IC50 = 86 nM T92144 CEQ1F2 24983299 IC50 = 2 nM T92144 C6JXE2 24983340 IC50 = 470 nM T92144 CK9TP6 24983359 IC50 = 250 nM T92144 CC39KU 24983384 IC50 = 310 nM T92144 C07PXL 24983399 IC50 = 590 nM T92144 C03XEW 24983494 IC50 = 110 nM T92144 CQ46VT 24983495 IC50 = 20 nM T92144 COB43M 25014810 IC50 = 340 nM T92144 CS96TK 25113168 IC50 = 4 nM T92144 CTV54O 25123227 IC50 > 10000 nM T92144 C1IYN7 25127854 IC50 > 1000 nM T92144 CKD14B 25127856 IC50 > 1000 nM T92144 CJBX60 25128180 IC50 > 1000 nM T92144 CC5SD9 25128181 IC50 > 1000 nM T92144 CQMU82 25138148 IC50 = 21 nM T92144 CD9O6K 25138149 IC50 = 93 nM T92144 CSO82D 25154877 Ki = 1160 nM T92144 CX0O5A 25178331 IC50 = 8900 nM T92144 C6FGQ1 25206346 IC50 = 840 nM T92144 CRO8T9 25263033 Ki > 2500 nM T92144 C41TLH 42603880 IC50 = 85000 nM T92144 CZ2VH7 42604008 IC50 = 95000 nM T92144 CU9E4P 42629114 IC50 > 10000 nM T92144 CJ5U1X 42639664 IC50 = 3.3 ug.mL-1 T92144 CTN41Y 44156909 IC50 = 840 nM T92144 CCFQ29 44187005 IC50 = 293 nM T92144 CEL61X 44229839 IC50 = 3200 nM T92144 CZFQ76 44291533 IC50 = 275 nM T92144 CEU2W4 44308690 IC50 = 150 nM T92144 CY6ZB5 44308830 IC50 = 7000 nM T92144 C1I6RG 44308968 IC50 = 239 nM T92144 C1I0LN 44308993 IC50 = 162 nM T92144 CKVZ38 44308994 IC50 = 970 nM T92144 CF9I2S 44309110 IC50 = 1020 nM T92144 C8VX1L 44309229 IC50 = 677 nM T92144 CZQ4S0 44309230 IC50 = 246 nM T92144 CHF28G 44309494 IC50 = 430 nM T92144 CYV2D7 44368815 IC50 = 6800 nM T92144 C7KZV2 44414322 IC50 = 17641 nM T92144 CJM06T 44414347 IC50 = 47793 nM T92144 CBY7D9 44414679 IC50 = 28 nM T92144 C0JF1Z 44414779 IC50 = 22 nM T92144 C7HQ1V 44418298 IC50 = 48 nM T92144 CO9H4N 44418299 IC50 = 4 nM T92144 CJF6B1 44418302 IC50 = 2 nM T92144 CYP61S 44418305 IC50 = 3 nM T92144 C6YW3N 44418309 IC50 = 3 nM T92144 C9W3GM 44418314 IC50 = 19 nM T92144 C3VD2Z 44418318 IC50 = 1 nM T92144 CT3N1H 44418321 IC50 = 5 nM T92144 CT12WM 44418327 IC50 = 2 nM T92144 C7J2XU 44418332 IC50 = 2 nM T92144 C7IO3E 44418339 IC50 = 2 nM T92144 CS25UA 44418346 IC50 = 2 nM T92144 CG49MW 44418350 IC50 = 6 nM T92144 CB1W8D 44418356 IC50 = 3 nM T92144 CN74KG 44418361 IC50 = 3 nM T92144 CAC8R3 44418362 IC50 = 7 nM T92144 C6W1LF 44418363 IC50 = 6 nM T92144 C01OZP 44418364 IC50 = 4 nM T92144 CM7OV4 44418365 IC50 = 4 nM T92144 CY8UZ5 44418366 IC50 = 8 nM T92144 CM9YH8 44418374 IC50 = 36 nM T92144 CZW1V5 44418379 IC50 = 29 nM T92144 C1DLQ9 44418386 IC50 = 20 nM T92144 C0NF4E 44418392 IC50 = 5 nM T92144 CVP5Q4 44418397 IC50 = 11 nM T92144 CT6ZD3 44418402 IC50 = 18 nM T92144 CLIY92 44418410 IC50 = 7 nM T92144 CFEA89 44418422 IC50 = 230 nM T92144 CLO5F6 44418448 IC50 = 4 nM T92144 CG5FS7 44418453 IC50 = 12 nM T92144 C1YGN9 44418460 IC50 = 10 nM T92144 C89MBJ 44418993 IC50 = 388 nM T92144 C31XOY 44418994 IC50 = 108 nM T92144 CRP04Z 44428103 IC50 = 1300 nM T92144 CBH1Y3 44433170 IC50 = 20000 nM T92144 C78NDQ 44433171 IC50 = 60 nM T92144 C13AMO 44433172 IC50 = 335 nM T92144 CDS5Q3 44433312 IC50 = 339 nM T92144 CVXH37 44433313 IC50 = 5500 nM T92144 C3MA7F 44433314 IC50 = 219 nM T92144 CJM89N 44433315 IC50 = 5370 nM T92144 C0UJZ7 44433316 IC50 = 3890 nM T92144 CIV7N0 44433317 IC50 = 437 nM T92144 C8WRS7 44433566 IC50 = 387 nM T92144 CT5W1U 44433567 IC50 = 1600 nM T92144 CKJ7I9 44433568 IC50 = 157 nM T92144 C0SI1L 44433569 IC50 = 82 nM T92144 CQ63SY 44433570 IC50 = 260 nM T92144 CZ29GV 44433571 IC50 = 78 nM T92144 CG91ZM 44433572 IC50 = 346 nM T92144 CG78NW 44433573 IC50 = 836 nM T92144 C8A4DV 44433574 IC50 = 250 nM T92144 CG4B9Z 44433575 IC50 = 1300 nM T92144 C65VKF 44433576 IC50 = 36 nM T92144 C4X7QS 44433577 IC50 = 40 nM T92144 CK4HC8 44433578 IC50 = 1500 nM T92144 C0C4QL 44433579 IC50 = 51 nM T92144 CONE50 44433580 IC50 = 59 nM T92144 CQWC12 44438817 IC50 = 46 nM T92144 CGV37F 44440254 IC50 = 40595 nM T92144 C5JUV3 44440256 IC50 = 13025 nM T92144 CFB56S 44440259 IC50 = 24747 nM T92144 CEW9G2 44440261 IC50 > 50000 nM T92144 CL52XP 44440291 IC50 = 13 nM T92144 CQX84Z 44440292 IC50 = 1 nM T92144 C35NRO 44440293 IC50 = 3 nM T92144 CZE89H 44440294 IC50 = 2 nM T92144 C2UG3R 44440295 IC50 = 5 nM T92144 CXD5L8 44440296 IC50 = 11 nM T92144 CK5UH6 44440297 IC50 = 6 nM T92144 CSBX36 44440298 IC50 = 4 nM T92144 CD81OT 44440299 IC50 = 55 nM T92144 C1HRG0 44440300 IC50 = 4 nM T92144 C1KN2U 44440301 IC50 = 6 nM T92144 CBH1R5 44440302 IC50 = 20 nM T92144 CPB2Z6 44440303 IC50 = 8 nM T92144 C6RC4L 44440304 IC50 = 17 nM T92144 CGN1Q4 44440305 IC50 = 9 nM T92144 CG5FA3 44447873 IC50 = 2 nM T92144 CM6A1T 44447874 IC50 = 148 nM T92144 CJ6T9P 44447875 IC50 = 264 nM T92144 CD20WZ 44447876 IC50 = 71 nM T92144 CPY39Q 44447877 IC50 = 23 nM T92144 C4JD3N 44447878 IC50 = 264 nM T92144 C2K6ZS 44447879 IC50 = 92 nM T92144 C2NMO0 44447881 IC50 = 28 nM T92144 CB2N8J 44447882 IC50 = 10 nM T92144 CSF9U6 44447883 IC50 = 93 nM T92144 C2BP9I 44447884 IC50 = 347 nM T92144 C9MPX0 44447885 IC50 = 300 nM T92144 C1M0DP 44447887 IC50 = 30 nM T92144 CTXY59 44447888 IC50 = 97 nM T92144 C4YMI9 44447890 IC50 = 30 nM T92144 C7L9AF 44447891 IC50 = 108 nM T92144 CHR96X 44447892 IC50 = 25 nM T92144 CZ8DG5 44447893 IC50 = 52 nM T92144 C5X2HE 44447894 IC50 = 23 nM T92144 CR65PM 44447895 IC50 = 26 nM T92144 CQH8F7 44447896 IC50 = 66 nM T92144 C3PH2E 44447897 IC50 = 46 nM T92144 CSB53H 44447898 IC50 = 45 nM T92144 CXL80U 44453148 IC50 = 726 nM T92144 C06KUB 44453149 IC50 = 83 nM T92144 CGA6S8 44453150 IC50 = 272 nM T92144 CMPZ16 44453151 IC50 = 300 nM T92144 C3DLE8 44453187 IC50 > 10000 nM T92144 CC6EP9 44453188 IC50 = 1000 nM T92144 CYS5W1 44453216 IC50 > 1000 nM T92144 C6E2SG 44453252 IC50 = 372 nM T92144 C6TMR8 44453253 IC50 = 1101 nM T92144 C4U7ZB 44453254 IC50 = 136 nM T92144 CQ9Y3M 44453489 IC50 = 5 nM T92144 CDV6X9 44454507 IC50 > 25000 nM T92144 C6SMY7 44454538 IC50 > 25000 nM T92144 CZI92T 44454651 IC50 > 25000 nM T92144 CIA39D 44454676 IC50 > 25000 nM T92144 C7DGA2 44454678 IC50 > 25000 nM T92144 C1F3LT 44454702 IC50 > 25000 nM T92144 CCW57R 44454703 IC50 > 25000 nM T92144 CFS7W2 44454728 IC50 > 25000 nM T92144 CTL43P 44454729 IC50 > 25000 nM T92144 CZC95J 44454731 IC50 > 25000 nM T92144 C7N2AQ 44473101 IC50 = 520 nM T92144 C4MG3F 44473102 IC50 = 24 nM T92144 CA85NJ 44473103 IC50 = 400 nM T92144 C0LY6E 44552561 EC50 = 300 nM T92144 C7KRU3 44552562 EC50 = 140 nM T92144 C3XTA7 44562721 Ki > 8300 nM T92144 C3Q0DX 44564789 IC50 = 1900 nM T92144 CP40XB 44564790 IC50 = 8600 nM T92144 C35NTB 44564791 IC50 = 8700 nM T92144 CJY83G 44564817 IC50 = 2500 nM T92144 CF2D1K 44564819 IC50 = 1300 nM T92144 C3CQ9K 44564820 IC50 > 10000 nM T92144 CI8V2L 44564821 IC50 > 10000 nM T92144 C9PO7J 44564860 IC50 = 4400 nM T92144 C16FJW 44564861 IC50 = 4100 nM T92144 C8AMX5 44564862 IC50 = 7000 nM T92144 CTR59U 44564863 IC50 > 10000 nM T92144 C9EY4C 44564864 IC50 > 10000 nM T92144 CG5Z7T 44564910 IC50 = 1000 nM T92144 CU9O4C 44564911 IC50 > 10000 nM T92144 CXZ15S 44564954 IC50 > 10000 nM T92144 CZ78WJ 44564955 IC50 > 10000 nM T92144 CJ1X9V 44565013 IC50 > 10000 nM T92144 CN2Q3D 44565014 IC50 = 4400 nM T92144 CM2GN3 44565015 IC50 = 1200 nM T92144 C14VTA 44581528 IC50 = 460 nM T92144 CM75ND 44581529 IC50 = 250 nM T92144 C6RJZ5 44581565 IC50 = 5 nM T92144 CE2C7W 44581602 IC50 = 240 nM T92144 CGQR60 44586767 IC50 > 100000 nM T92144 CVRQ96 44586768 IC50 = 68000 nM T92144 C05HTO 44586769 IC50 = 11000 nM T92144 CX0R8V 44586770 IC50 = 41000 nM T92144 CQA2K1 44586794 IC50 = 27000 nM T92144 CH67VY 44586829 IC50 > 100000 nM T92144 C0HOF8 44586830 IC50 = 5200 nM T92144 COI0E3 44586831 IC50 = 83000 nM T92144 C86ADQ 44586832 IC50 = 64000 nM T92144 CZAF65 44586833 IC50 > 100000 nM T92144 CWP37F 44586834 IC50 = 5600 nM T92144 CT5HM0 44586867 IC50 = 2900 nM T92144 CGK6C7 44586868 IC50 > 100000 nM T92144 C70DAO 44586869 IC50 = 370 nM T92144 C2JIZ9 44586870 IC50 > 100000 nM T92144 CZM16E 44586871 IC50 = 68000 nM T92144 CYU2G3 44586896 IC50 = 21000 nM T92144 C7G6KH 44586897 IC50 = 2800 nM T92144 C4L9BF 44586898 IC50 > 100000 nM T92144 CM45ZR 44586899 IC50 > 100000 nM T92144 CVU93G 44586900 IC50 > 100000 nM T92144 CMV3W2 44586901 IC50 > 100000 nM T92144 CV2W4P 44586928 IC50 > 100000 nM T92144 C95XRW 44586929 IC50 > 100000 nM T92144 CCT91D 44586930 IC50 = 6400 nM T92144 CJ4HT0 44587324 IC50 > 100000 nM T92144 CD56YX 44587325 IC50 > 100000 nM T92144 C4KW0O 44587326 IC50 = 14000 nM T92144 CR80YC 45375946 IC50 = 440 nM T92144 C6E2SC 45482700 IC50 > 10000 nM T92144 CZXH74 45482750 IC50 > 10000 nM T92144 CH5VI6 46186825 IC50 = 75 nM T92144 CUA97D 46209401 IC50 = 740 nM T92144 C8YPN0 46225596 IC50 = 230 nM T92144 C34JTS 46225597 IC50 = 330 nM T92144 CGD73B 46225598 IC50 = 590 nM T92144 C3E0PU 46225599 IC50 = 360 nM T92144 CRDY89 46225610 EC50 = 10000 nM T92144 C0JMT8 46225611 IC50 = 390 nM T92144 CF0D5J 46225612 IC50 = 54 nM T92144 CFVO38 46225632 IC50 = 3100 nM T92144 CLZ1O6 46225634 EC50 = 2100 nM T92144 C07VDX 46225635 IC50 = 670 nM T92144 CT70DX 46225640 IC50 = 68 nM T92144 CJUF68 46225641 IC50 = 510 nM T92144 C6AJ5N 46225647 IC50 = 235 nM T92144 C2WCV1 46225648 IC50 = 4000 nM T92144 CBS96A 46225649 IC50 > 10000 nM T92144 C38BFC 46225657 IC50 = 110 nM T92144 CD0A6F 46225658 IC50 = 350 nM T92144 C1B3KS 46225663 IC50 = 9 nM T92144 CU46XI 46225664 IC50 = 410 nM T92144 CO3HS2 46225665 IC50 = 510 nM T92144 C2UV1S 46225666 IC50 = 3300 nM T92144 CX5B1G 46225667 IC50 = 615 nM T92144 C2Q9OH 46225668 IC50 > 10000 nM T92144 CM14FH 46225680 IC50 = 880 nM T92144 CQS96E 46225681 IC50 = 6100 nM T92144 CJIK35 46225682 IC50 = 1400 nM T92144 C8S4QA 46225688 IC50 = 38 nM T92144 CYZV41 46231219 IC50 = 1567 nM T92144 C7J5UP 46231220 IC50 = 3961 nM T92144 CC96GZ 46231221 IC50 = 2367 nM T92144 C40JIK 46836783 IC50 = 76 nM T92144 C18YZM 46836784 IC50 = 27 nM T92144 CL2YG9 46836785 IC50 = 166 nM T92144 C0GA7Y 46836852 IC50 > 3000 nM T92144 CL1E8Y 46836853 IC50 > 3000 nM T92144 CF5J7R 46836854 IC50 = 10 nM T92144 CRQ61H 46836855 IC50 > 3000 nM T92144 C2DB9U 46836856 IC50 = 4 nM T92144 CX93NC 46836917 IC50 > 1000 nM T92144 CL9N5J 46879815 IC50 = 70 nM T92144 CFU29R 46879816 IC50 = 340 nM T92144 CX0B4D 46879872 IC50 = 490 nM T92144 C8V7LX 46879873 IC50 = 370 nM T92144 CHL36R 46889321 IC50 = 102 nM T92144 CA9J0L 46889322 IC50 = 469 nM T92144 COI7R4 46889323 IC50 = 9 nM T92144 CR8VH5 46889324 IC50 = 17 nM T92144 CJZC67 46889343 IC50 = 27 nM T92144 CZI7F3 46889344 IC50 = 16 nM T92144 CVK8I9 46889345 IC50 = 142 nM T92144 CVJ9X5 46889346 IC50 = 715 nM T92144 CTJ6L7 46889382 IC50 = 554 nM T92144 C4W7IC 46889383 IC50 = 88 nM T92144 C83AHJ 46889384 IC50 = 24 nM T92144 C9PZ4W 46889385 IC50 = 103 nM T92144 CGYT07 46889401 IC50 = 53 nM T92144 CMT73H 46889402 IC50 = 18 nM T92144 CAZ69B 46889403 IC50 = 300 nM T92144 CKP3D5 46889404 IC50 = 350 nM T92144 CB7SP1 46889850 IC50 = 44 nM T92144 CN19IK 46889851 IC50 = 41 nM T92144 CSQF75 46889884 IC50 = 14 nM T92144 CH8KA5 46889885 IC50 = 3 nM T92144 CP56KX 46889886 IC50 = 10 nM T92144 CW7AR1 46889887 IC50 = 10 nM T92144 CMNK35 46889911 IC50 = 3 nM T92144 CHW3Z2 46889912 IC50 = 21 nM T92144 CIV0K1 46889913 IC50 = 78 nM T92144 CST80X 46889914 IC50 = 41 nM T92144 CM02UJ 46890253 IC50 = 1 nM T92144 CB7VI8 46890254 IC50 = 82 nM T92144 C7V3IA 46890314 IC50 = 215 nM T92144 CHE6A1 46890315 IC50 = 248 nM T92144 C60GAV 46929544 IC50 = 630 nM T92144 CHSF07 49806372 IC50 > 1000 nM T92144 CD2K4R 50908681 Ki > 1000000 nM T92144 CM42BY 51000510 Ki > 1000000 nM T92144 CEQN27 52936621 Ki > 1000 nM T92144 C8NA4L 53384644 IC50 = 50000 nM T92144 CM8JX1 56604907 IC50 = 100 nM T92144 CR50TJ 56835147 IC50 > 10000 nM T92144 CGLH06 56950183 IC50 = 241 nM T92144 CE59QS 57505507 IC50 > 1000 nM T92144 C8P6RD 57505528 IC50 = 5100 nM T92144 CT3EW2 59292007 IC50 > 1000 nM T92144 CXJ63M 59603829 IC50 = 4700 nM T92144 CQEU96 59603842 IC50 = 660 nM T92144 C1MR8Q 60097495 IC50 > 1000 nM T92144 C9A1YD 67218825 IC50 = 8.8 nM T92144 CF7ZV0 67219275 IC50 > 10000 nM T92144 C1V7FU 67219433 IC50 = 45 nM T92144 CNE0Z2 67219498 IC50 = 345 nM T92144 CN1FG6 67219570 IC50 = 12 nM T92144 C4AV2K 67219622 IC50 = 423 nM T92144 CT0V2G 67219629 IC50 = 745 nM T92144 CA63QI 67219716 IC50 = 361 nM T92144 CV63UL 67240318 IC50 > 10000 nM T92144 C5DGR9 69036886 IC50 = 1040 nM T92144 CAOE64 69412987 IC50 = 9750 nM T92144 C38MXT 70693454 IC50 = 22 nM T92144 CEBO91 71452977 IC50 > 10000 nM T92144 CZ31PU 71583657 IC50 > 10000 nM T92144 C6R8DI 72943374 IC50 = 208 nM T92144 CWC19I 73355703 IC50 = 95 nM T92144 C6UA4K 73356522 IC50 = 137 nM T92144 CPG3A5 86302574 IC50 > 30000 nM T92144 C1HW4B 89735655 IC50 > 100000 nM T92144 CMH6T8 90664306 IC50 = 120 nM T92144 C3KLI5 118723185 IC50 > 100000 nM T92144 CUO0C5 132156633 IC50 > 10000 nM T92144 CK9D4A 135428921 IC50 = 120 nM T92144 C16XLU 135454992 IC50 = 1000 nM T92144 C64EMD 135500075 IC50 = 180 nM T92144 CVZ08D 135509841 IC50 = 400 nM T92144 C0J3BN 135678111 IC50 = 23273 nM T92144 C2PAV1 135971426 IC50 = 5300 nM T92144 CXC69T 137321158 IC50 = 75 nM T92144 C9UW0D 137632355 IC50 = 2.47 nM T92144 CQ7MZ6 137633392 IC50 = 0.6 nM T92144 CSQ87K 137634450 IC50 = 6.34 nM T92144 CKL1S0 137635182 IC50 > 1000 nM T92144 C9F5GA 137636582 IC50 = 9.68 nM T92144 C6ESL5 137638961 IC50 > 1000 nM T92144 CX95WZ 137639923 IC50 > 1000 nM T92144 CBGR42 137641572 IC50 = 0.13 nM T92144 CP5Q4H 137642451 IC50 = 13.22 nM T92144 CWB74C 137642729 IC50 = 87.38 nM T92144 C4DRX1 137643187 IC50 = 510 nM T92144 CPE93W 137643241 IC50 = 15.68 nM T92144 CAY1L6 137645294 IC50 > 1000 nM T92144 C6DOB5 137645672 IC50 = 1.95 nM T92144 CPI1C6 137646147 IC50 = 1.14 nM T92144 CN5R6A 137646618 IC50 = 52.04 nM T92144 CVZ85B 137647227 IC50 = 3.49 nM T92144 CYH05X 137652479 IC50 = 49.97 nM T92144 C19AQU 137654195 IC50 = 6.05 nM T92144 C1HT8J 137654707 IC50 = 904.52 nM T92144 C1Q7UO 137657235 IC50 = 134.12 nM T92144 C2M6IZ 137657987 IC50 = 0.16 nM T92144 C2VRD0 137658292 IC50 = 164.35 nM T92144 C8E4QA 137658885 IC50 = 23.78 nM T92144 CZT18Q 137661519 IC50 = 6.72 nM T92144 COCU58 141538430 IC50 = 5.46 nM T92144 C6Y5NP 145949388 IC50 = 98.12 nM T92144 CB3Z1W 145949428 IC50 = 5.63 nM T92144 CYEK37 145949698 IC50 = 59.93 nM T92144 CGB21E 145949773 IC50 = 21.2 nM T92144 CVTZ73 145950013 IC50 = 54.9 nM T92144 C3Q1CR 145950413 IC50 > 500 nM T92144 CKU2J6 145951459 IC50 = 16.55 nM T92144 CO0KI7 145951584 IC50 = 10.29 nM T92144 CWUM46 145952127 IC50 = 133.47 nM T92144 CS5FN6 145952182 IC50 = 31.15 nM T92144 CL1J3N 145952225 IC50 = 105.07 nM T92144 C0U2SX 145952427 IC50 = 134.67 nM T92144 C1C2KL 145952546 IC50 = 16.77 nM T92144 C1KX3F 145952675 IC50 = 14.49 nM T92144 CWU7J4 145952685 IC50 = 37.24 nM T92144 CY3M1A 145952761 IC50 = 21.27 nM T92144 CETX79 145953187 IC50 = 22.15 nM T92144 CQO92P 145953233 IC50 = 4.85 nM T92144 C6WB5A 145953633 IC50 = 97.74 nM T92144 C09BOY 145953698 IC50 = 64.33 nM T92144 C8K3IT 145953806 IC50 > 500 nM T92144 CN59EV 145954386 IC50 > 500 nM T92144 CX94IY 145954428 IC50 = 3.59 nM T92144 C5Z3NW 145954580 IC50 = 28.32 nM T92144 CHBA54 145954987 IC50 = 12.81 nM T92144 C4CQI1 145955346 IC50 > 500 nM T92144 CFC1R5 145955514 IC50 = 14.2 nM T92144 CZ1X4T 145956589 IC50 = 73.59 nM T92144 C1Z5BV 145956656 IC50 = 21.52 nM T92144 C5VSC7 145956704 IC50 = 2.13 nM T92144 C0Y2TV 145956729 IC50 = 90.86 nM T92144 CJ4F8V 145956840 IC50 = 68.68 nM T92144 CPG5X6 145957058 IC50 = 24.75 nM T92144 CA72LX 145957228 IC50 = 7.97 nM T92144 C7YBO3 145957370 IC50 = 432.35 nM T92144 CZ6O9G 145957666 IC50 = 14.2 nM T92144 CB4P3U 145957792 IC50 > 500 nM T92144 CMSE06 145957839 IC50 > 500 nM T92144 CZM5L3 145959497 IC50 = 14.65 nM T92144 CVZ4Q2 145959877 IC50 = 88.64 nM T92144 CH3YK9 145960253 IC50 > 500 nM T92144 CA9LY3 145960784 IC50 = 42.15 nM T92144 C1U6NF 145961006 IC50 = 245.28 nM T92144 CMZN84 145961642 IC50 > 500 nM T92144 CCK21X 145962292 IC50 = 115.15 nM T92144 CY7B2V 145962703 IC50 = 65.26 nM T92144 CR75NT 145963742 IC50 = 13.75 nM T92144 C8YM3U 145971698 IC50 > 500 nM T92144 CBI6C0 145971699 IC50 = 16.7 nM T92144 CAR6T3 145971936 IC50 = 19.8 nM T92144 CDB5N6 145972176 IC50 = 9.19 nM T92144 C8S6VJ 145972201 IC50 = 9.77 nM T92144 CZ5P0E 145972710 IC50 > 500 nM T92144 CC1F9L 147598461 IC50 = 51.86 nM T92144 CS8BJ7 149949125 IC50 > 1000 nM T92144 CV6A7T 149961985 IC50 = 265.72 nM T92144 CJL17Q 150336955 IC50 = 9.11 nM T92144 C6PG4T 150482255 IC50 > 1000 nM T92144 CP9JW5 150533442 IC50 = 0.82 nM T92144 C2K9BQ 150746217 IC50 > 1000 nM T92144 CHXZ94 151105657 IC50 > 1000 nM T92144 CU7T8Y 151363744 IC50 > 1000 nM T92144 C90NHE 151428103 IC50 = 1.79 nM T92144 CFE6I9 152015157 IC50 = 51.44 nM T92144 C24QHN 152058632 IC50 = 46.39 nM T92144 CJ4G3V 152221091 IC50 = 77.42 nM T92144 CJSM72 152346156 IC50 = 0.36 nM T92144 CZ7GT5 152346369 IC50 = 2.69 nM T92144 CRE82P 155510352 IC50 = 13.71 nM T92144 C2MD1Q 155513187 IC50 > 10000 nM T92144 C83CSB 155515100 IC50 = 0.73 nM T92144 C98MWS 155518832 IC50 = 0.28 nM T92144 CT6V3O 155519533 IC50 = 210 nM T92144 C6CPO5 155520481 IC50 > 1000 nM T92144 CU6Z5O 155520650 IC50 = 480 nM T92144 C7QM2L 155520700 IC50 > 1000 nM T92144 CTC34D 155520839 IC50 = 0.26 nM T92144 CD2YM4 155523255 IC50 = 25.74 nM T92144 CBP7G1 155524105 IC50 = 61.26 nM T92144 CV9Y3X 155527350 IC50 = 5.45 nM T92144 CXY94L 155534355 IC50 > 1000 nM T92144 C9P3ON 155542000 IC50 > 1000 nM T92144 CP4KT1 155544904 IC50 = 0.3 nM T92144 CDKF14 155556917 IC50 = 24.19 nM T92144 C3BPZ9 155557063 IC50 > 1000 nM T92144 C40IYS 155562258 IC50 = 26.3 nM T92144 C81JZW 155563388 IC50 = 1390 nM T92144 CFG6Z5 155564309 IC50 = 0.45 nM T92144 D02BXJ 46864270 IC50 = 2.2 nM T92144 D04ZWF 53396311 IC50 > 5000 nM T92144 D06QWO 14824655 IC50 > 10 ug.mL-1 T92144 D06WGX 9549184 IC50 > 50000 nM T92144 D07AIB 712152 IC50 = 17870 nM T92144 D07OXC 11650194 IC50 = 285 nM T92144 D0A1CM 5281855 IC50 = 260 nM T92144 D0BS6R 9549183 IC50 = 1484 nM T92144 D0D6DH 10125830 IC50 > 50000 nM T92144 D0D6MH 11617559 IC50 > 20000 nM T92144 D0EE6A 6398883 IC50 > 10000 nM T92144 D0G3SZ 6918469 IC50 = 9.8 ug.mL-1 T92144 D0GN5Z 5281295 IC50 = 950 nM T92144 D0IR6U 5494425 IC50 = 24000 nM T92144 D0L0HG 766949 IC50 > 10000 nM T92144 D0N3JX 44433173 IC50 = 114 nM T92144 D0OZ2S 11785878 IC50 = 750 nM T92144 D0Q3KS 9957049 IC50 > 25000 nM T92144 D0R2WK 16038120 EC50 = 1167 nM T46685 D0E3TC 44259 IC50 = 14.2 nM T46685 D00OWF 5280953 IC50 = 26 nM T46685 D00PWQ 3820 IC50 > 10000 nM T46685 D05BVP 3232621 IC50 = 59 nM T46685 D06MBI 1893668 IC50 = 17 nM T46685 D09CDR 77105816 IC50 = 23 nM T46685 D0CC7E 77105818 IC50 = 23 nM T46685 D0JQ0Z 46916176 IC50 = 173 nM T46685 D0PO8N 117881270 IC50 = 300 nM T46685 D0Q3VZ 135398522 IC50 = 71 nM T46685 D0WX0K 71680628 IC50 = 71 nM T46685 C8HN2C 3798 IC50 >= 10000 nM T46685 CVJC65 398318 IC50 > 10000 nM T46685 CFBU18 400433 IC50 = 530 nM T46685 C3K9FJ 401171 IC50 = 120 nM T46685 CN6AY0 491467 IC50 > 10000 nM T46685 C7XM8E 621030 IC50 > 10000 nM T46685 C3D1HC 762415 IC50 > 10000 nM T46685 CIW3E8 939111 IC50 = 210 nM T46685 CFA92X 1237489 IC50 = 7520 nM T46685 CD1A9T 1241605 IC50 = 5700 nM T46685 C2EUG6 1474849 IC50 > 10000 nM T46685 CKNV93 2808989 IC50 > 10000 nM T46685 CP38YL 2823823 IC50 = 4500 nM T46685 CU80LI 3233012 IC50 = 22 nM T46685 CW4C3P 3235048 IC50 = 4805 nM T46685 CGAT36 5327151 IC50 = 868 nM T46685 C2TVO1 5328202 IC50 > 10000 nM T46685 CFW19M 5329009 IC50 = 7600 nM T46685 CLM7V5 5371900 IC50 = 10000 nM T46685 CZU0A4 5479542 IC50 >= 10000 nM T46685 CO6KI2 5930298 IC50 > 10000 nM T46685 CLN2G8 6475560 IC50 = 8300 nM T46685 C0MGV7 7048595 IC50 = 1500 nM T46685 C14UAT 7574840 IC50 > 10000 nM T46685 CL80ZW 9863168 IC50 > 10000 nM T46685 C3DM8P 11221000 IC50 >= 10000 nM T46685 C4HUM2 11232168 IC50 > 10000 nM T46685 C81HMZ 11242728 IC50 > 10000 nM T46685 CP04JC 11666231 IC50 = 200 nM T46685 CPI54D 11953235 EC50 = 48000 nM T46685 CJ0NW4 12235681 IC50 = 60 nM T46685 CIDQ65 12248890 IC50 > 10000 nM T46685 CR3BS0 12248905 IC50 = 170 nM T46685 CX27EP 13975510 IC50 = 4370 nM T46685 CJ35KT 16751570 IC50 = 1400 nM T46685 CMW42V 19079253 IC50 = 3600 nM T46685 CC9V2Y 24882562 IC50 = 93 nM T46685 CWIE80 25190906 IC50 = 190 nM T46685 CJ9I2T 25190908 IC50 = 680 nM T46685 CGLQ20 44223952 IC50 = 96 nM T46685 CR6VH2 44223953 IC50 = 69 nM T46685 C2IBW0 44223954 IC50 = 931 nM T46685 CS3Q2Y 44223955 IC50 = 90 nM T46685 C5M1UN 44223957 IC50 = 98 nM T46685 CK8G1T 44223965 IC50 = 130 nM T46685 CJ8KD4 44223966 IC50 = 39 nM T46685 CCW0V4 44223967 IC50 = 191 nM T46685 CF78WD 44223968 IC50 = 888 nM T46685 CNE30X 44223970 IC50 = 20 nM T46685 CYR45S 44223971 IC50 = 28 nM T46685 CLZ62P 44223973 IC50 = 11 nM T46685 CIXB09 44223974 IC50 = 86 nM T46685 C2OBX8 44223977 IC50 = 111 nM T46685 C3VRO9 44557921 IC50 > 10000 nM T46685 C3HW7L 44570553 IC50 > 30000 nM T46685 C17PVE 44570554 IC50 > 30000 nM T46685 CLOY92 44570599 IC50 = 15000 nM T46685 CK06LT 44570600 IC50 = 3000 nM T46685 C3JBN1 44968184 IC50 = 89 nM T46685 CYW79D 44968186 IC50 = 14 nM T46685 C5OYK3 44968199 IC50 = 798 nM T46685 C2T0EM 44968221 IC50 = 2083 nM T46685 C8NA2J 44968224 IC50 = 899 nM T46685 CR8DC5 44968225 IC50 = 480 nM T46685 CV19YK 44968230 IC50 = 206 nM T46685 CD4ZN1 44968231 IC50 = 1522 nM T46685 C16QFN 46172966 IC50 = 5459 nM T46685 CB32ET 46172972 IC50 > 10000 nM T46685 CN26HW 46172980 IC50 = 76 nM T46685 CGH05O 46172984 IC50 = 277 nM T46685 C15EJK 46916169 IC50 = 1561 nM T46685 CHG8C4 46916170 IC50 = 176 nM T46685 CI56BA 46916172 IC50 = 128 nM T46685 CZ5DJ4 46916177 IC50 = 192 nM T46685 CXK37B 46916178 IC50 = 522 nM T46685 CL1GW0 46916179 IC50 = 227 nM T46685 CZ6DK4 46916182 IC50 = 598 nM T46685 CK7PM2 46918486 IC50 > 10000 nM T46685 C8BQ1W 46926509 IC50 > 10000 nM T46685 CCUG10 46926515 IC50 = 102 nM T46685 C9NC6W 46926516 IC50 = 34 nM T46685 CZ1D2A 46926518 IC50 = 11 nM T46685 C7S6HT 46926519 IC50 = 16 nM T46685 CG1K5A 46926520 IC50 = 626 nM T46685 CVF48X 46926521 IC50 = 180 nM T46685 C4ULH5 46926522 IC50 = 13 nM T46685 CPE98Z 46926523 IC50 = 8 nM T46685 C6WLX1 46926524 IC50 = 2370 nM T46685 C61LUI 46926526 IC50 = 1262 nM T46685 C0IVD1 46926527 IC50 = 24 nM T46685 CE4SU5 47298428 IC50 = 500 nM T46685 CAYI59 49795862 IC50 = 183 nM T46685 C1UQN4 49795863 IC50 = 1783 nM T46685 CU8OC0 49795864 IC50 = 1598 nM T46685 C7T5HW 49795865 IC50 = 73 nM T46685 C6N8EY 49795866 IC50 = 41 nM T46685 C7XS1Z 49795867 IC50 = 964 nM T46685 C6VQ7Y 49853605 IC50 = 2300 nM T46685 C20IFM 49854737 IC50 = 2000 nM T46685 CXI39D 49854741 IC50 = 1700 nM T46685 C4D3JF 49854742 IC50 = 3000 nM T46685 C5W3DH 49854744 IC50 = 1300 nM T46685 C9I4LQ 49855059 IC50 = 4000 nM T46685 C5EWG8 49855158 IC50 = 16 nM T46685 CD2K4R 50908681 Ki > 1000000 nM T46685 CBH27E 53361525 IC50 = 65 nM T46685 C9EKT8 53361563 IC50 = 32 nM T46685 C73OJM 53361564 IC50 = 42 nM T46685 CB4U8E 53361565 IC50 = 41 nM T46685 CP1K6C 53361566 IC50 = 80 nM T46685 CJG68X 53361567 IC50 = 26 nM T46685 C49CKH 53362267 IC50 = 2300 nM T46685 CY9FK8 53362270 IC50 = 1300 nM T46685 C14ZTR 53362271 IC50 > 10000 nM T46685 C6SCG9 53362272 IC50 > 10000 nM T46685 CXQ85R 53362273 IC50 = 1500 nM T46685 CDRI60 53362320 IC50 = 1300 nM T46685 CE27PN 53362321 IC50 = 2500 nM T46685 C0JI6Z 53362322 IC50 = 2300 nM T46685 CBF85Z 53362323 IC50 = 870 nM T46685 C18ZQY 53362378 IC50 = 180 nM T46685 C3SXT4 53362379 IC50 = 1500 nM T46685 C8LT5F 53362380 IC50 = 1600 nM T46685 CW7XG8 53362381 IC50 = 1800 nM T46685 C2DTF5 53362382 IC50 = 380 nM T46685 C5UH7N 53363043 IC50 = 380 nM T46685 CA2DU1 53363044 IC50 = 70 nM T46685 CL5K0B 53363045 IC50 = 7100 nM T46685 CDYX16 53363046 IC50 = 120 nM T46685 CUFT73 53363047 IC50 = 67 nM T46685 C9THC6 53363128 IC50 = 1000 nM T46685 CW9C6N 53363129 IC50 = 610 nM T46685 C6XMD8 53363219 IC50 = 30 nM T46685 CS6N8Z 54581884 IC50 = 6164 nM T46685 CUP75Y 54582100 IC50 > 10000 nM T46685 CA0B2E 54585955 IC50 > 10000 nM T46685 CDIE71 56662956 IC50 = 750 nM T46685 CSE8X0 56662957 IC50 = 87 nM T46685 CF4H1O 56683277 IC50 > 10000 nM T46685 CP2KW6 56683332 IC50 = 530 nM T46685 CZ1AP7 56956644 IC50 = 1400 nM T46685 CT6XL0 57466811 IC50 = 118 nM T46685 CVTB94 58047131 IC50 = 100 nM T46685 C3ZPO8 58880668 IC50 > 10000 nM T46685 CW9AE7 60034150 EC50 = 22000 nM T46685 CV63UL 67240318 IC50 > 10000 nM T46685 CF87LR 71449511 IC50 = 5200 nM T46685 C6D2SK 71449512 IC50 > 10000 nM T46685 C34UIP 71451312 IC50 > 10000 nM T46685 CQ6GO1 71453130 IC50 = 3400 nM T46685 C5OM3N 71453131 IC50 > 10000 nM T46685 CXM3F7 71453132 IC50 > 10000 nM T46685 CK3GE4 71454861 IC50 = 2100 nM T46685 C9WPB8 71456635 IC50 > 10000 nM T46685 C1XLB9 71456636 IC50 > 10000 nM T46685 C96MVO 71456637 IC50 > 10000 nM T46685 CHZK01 71458489 IC50 > 10000 nM T46685 CJA07E 71458490 IC50 > 10000 nM T46685 CJF7O0 71460338 IC50 = 3300 nM T46685 CC9A3B 71460339 IC50 = 2200 nM T46685 CK5Z0O 71462038 IC50 > 10000 nM T46685 C5JHL1 71462039 IC50 > 10000 nM T46685 C3FI8H 71462040 IC50 > 10000 nM T46685 CVIA91 71553085 IC50 = 3450 nM T46685 C1TR3O 71553152 IC50 = 11210 nM T46685 CXTW04 71568938 IC50 = 410 nM T46685 C07WEJ 71568939 IC50 > 10000 nM T46685 C86MGW 71568941 IC50 > 10000 nM T46685 CK34WJ 71568942 IC50 = 1500 nM T46685 C8I3YN 71568943 IC50 > 10000 nM T46685 CC2R7D 71568945 IC50 > 10000 nM T46685 C7Z2GN 71569099 IC50 = 2000 nM T46685 CAZ32T 71569100 IC50 > 10000 nM T46685 C12ECZ 71569101 IC50 > 10000 nM T46685 CA8GX1 71569102 IC50 > 10000 nM T46685 CG0K8R 71569103 IC50 > 10000 nM T46685 C83ICT 71569104 IC50 > 10000 nM T46685 C6A0NQ 71569105 IC50 = 4200 nM T46685 C6Q7GK 71569254 IC50 > 10000 nM T46685 C5FN7Z 71569255 IC50 > 10000 nM T46685 C5R6PE 71569256 IC50 > 10000 nM T46685 C6RXK0 71569257 IC50 > 10000 nM T46685 CLE2Y1 71569258 IC50 > 10000 nM T46685 C7BL0Y 71569259 IC50 > 10000 nM T46685 C8C6FB 71569260 IC50 > 10000 nM T46685 C0I5SQ 71569413 IC50 > 10000 nM T46685 CQ6DF7 71569414 IC50 > 10000 nM T46685 CO04JY 71569415 IC50 > 10000 nM T46685 CXQ3O2 71569416 IC50 > 10000 nM T46685 CE49AB 71569417 IC50 > 10000 nM T46685 C3BUI6 71569418 IC50 > 10000 nM T46685 CRB13S 71569419 IC50 > 10000 nM T46685 CZ3CP7 71569420 IC50 > 10000 nM T46685 CXKT34 71569578 IC50 > 10000 nM T46685 CR7G9C 71569579 IC50 = 2800 nM T46685 C0BCN8 71569580 IC50 = 5100 nM T46685 CSB86F 71569581 IC50 > 10000 nM T46685 CLS70D 71569582 IC50 > 10000 nM T46685 C0V9UZ 71569583 IC50 = 680 nM T46685 C53IRH 71569584 IC50 > 10000 nM T46685 CV25GR 71569755 IC50 > 10000 nM T46685 CR78SP 71569756 IC50 > 10000 nM T46685 CM0CU6 71569757 IC50 > 10000 nM T46685 C5D8XE 71569758 IC50 = 3100 nM T46685 C1U2MX 71569759 IC50 = 6100 nM T46685 CP2RM4 71569760 IC50 > 10000 nM T46685 CI76UG 71569761 IC50 > 10000 nM T46685 C2NQG6 71569908 IC50 > 10000 nM T46685 CF67VW 71569909 IC50 > 10000 nM T46685 C2N1KZ 71569910 IC50 = 1600 nM T46685 C2R0ZU 71569911 IC50 = 2300 nM T46685 CZ9RS8 71569912 IC50 > 10000 nM T46685 CL3CP9 71569913 IC50 = 6800 nM T46685 COX8D5 71569914 IC50 > 10000 nM T46685 C8I6BH 71570062 IC50 = 790 nM T46685 C19FHW 71719163 IC50 > 10000 nM T46685 C1J8CH 71719164 IC50 > 10000 nM T46685 CDUS45 72725107 IC50 = 690 nM T46685 C2BK6U 72725108 IC50 = 610 nM T46685 CW2AL3 72725109 IC50 > 10000 nM T46685 CLW7C4 72725110 IC50 = 1000 nM T46685 CL9X7G 72725111 IC50 > 10000 nM T46685 CC6Q8Y 72725113 IC50 = 49 nM T46685 CWPD50 72725173 IC50 = 320 nM T46685 C0ZQT7 72725176 IC50 > 10000 nM T46685 CK43OC 72725177 IC50 > 10000 nM T46685 C03EJC 72725178 IC50 > 10000 nM T46685 CJ1IA8 72725179 IC50 > 10000 nM T46685 CWX65J 72725233 IC50 > 10000 nM T46685 CMN12Z 72725234 IC50 > 10000 nM T46685 C6RHQ4 72725235 IC50 > 10000 nM T46685 CGDC83 72725236 IC50 > 10000 nM T46685 CIJC97 72725237 IC50 > 10000 nM T46685 C4BV9L 73426232 EC50 > 1000000 nM T46685 CM0Y4P 74762666 EC50 = 800 nM T46685 C89QWD 76309937 IC50 > 10000 nM T46685 C63KPU 76313653 IC50 > 10000 nM T46685 C0A5UJ 76313654 IC50 > 10000 nM T46685 CA09CK 76331770 IC50 > 10000 nM T46685 C5P9AJ 76335356 IC50 > 10000 nM T46685 C2K8WN 76335357 IC50 > 10000 nM T46685 CFT3M1 76335358 IC50 > 10000 nM T46685 C3FZN9 76335359 IC50 > 10000 nM T46685 CJ8KR4 76335360 IC50 > 10000 nM T46685 CWQA01 76335361 IC50 > 10000 nM T46685 C21JAS 76853169 IC50 = 830 nM T46685 CW64MP 77105434 IC50 = 1500 nM T46685 CU04XY 77105624 IC50 = 230 nM T46685 C3NX4F 77105815 IC50 = 56 nM T46685 CEW7R1 77105817 IC50 = 1600 nM T46685 CIM47W 77105819 IC50 = 1600 nM T46685 CTIA65 77105820 IC50 = 2400 nM T46685 CH79MO 77105821 IC50 = 1400 nM T46685 CKB1P9 77106023 IC50 = 41 nM T46685 CTP6N7 77106024 IC50 > 10000 nM T46685 CXYW85 77106025 IC50 = 230 nM T46685 C2UDS0 77106026 IC50 = 620 nM T46685 C97SJD 77106027 IC50 = 570 nM T46685 CFQ10R 77106028 IC50 = 51 nM T46685 CO14DP 77106030 IC50 = 34 nM T46685 C5GM2W 77106233 IC50 = 2900 nM T46685 C9G3PA 77106234 IC50 = 430 nM T46685 CPD27I 77106235 IC50 = 47 nM T46685 CLOR37 77106236 IC50 = 86 nM T46685 C2GLD8 77106237 IC50 = 160 nM T46685 C8D3XO 86765295 IC50 = 7000 nM T46685 C0GYK1 86765296 IC50 = 170 nM T46685 CB40PI 90306552 IC50 > 10000 nM T46685 CUY63S 90645193 IC50 > 10000 nM T46685 C0Y8ZK 91933875 IC50 > 10 nM T46685 C3KJ8R 98073446 IC50 = 19.7 nM T46685 CE3LO6 102490713 IC50 = 88 nM T46685 CJ50DW 102490714 IC50 = 2500 nM T46685 C7WEL6 102490715 IC50 = 280 nM T46685 CKZA09 102490716 IC50 = 1100 nM T46685 CT97XD 102490717 IC50 = 690 nM T46685 C5W3ZK 102490718 IC50 = 2400 nM T46685 C8G5IT 118714396 IC50 = 100 nM T46685 CB8G1T 118714397 IC50 = 1900 nM T46685 CEB3G4 118714398 IC50 = 2000 nM T46685 CTUZ03 118714399 IC50 = 2100 nM T46685 CRV8H7 118714400 IC50 = 300 nM T46685 C7PAU6 118714401 IC50 = 1000 nM T46685 C6FQ8M 118714402 IC50 = 50 nM T46685 CJ89SC 118714404 IC50 = 50 nM T46685 C1GU9B 118714405 IC50 = 300 nM T46685 CF2IE6 118714406 IC50 = 400 nM T46685 C2ZBH0 118714407 IC50 = 200 nM T46685 CK64OD 118714410 IC50 = 1900 nM T46685 CY19HB 118731162 IC50 = 1700 nM T46685 CJH4V3 118731163 IC50 = 130 nM T46685 CU7QB1 118731164 IC50 = 110 nM T46685 CC8JB6 118731165 IC50 = 190 nM T46685 CT0C1Y 118731166 IC50 = 71 nM T46685 C0VG9C 118731167 IC50 = 910 nM T46685 CE09BY 118731168 IC50 = 500 nM T46685 C2G8WI 118731169 IC50 = 520 nM T46685 C8RP0D 118731170 IC50 = 180 nM T46685 CCJ12T 118731171 IC50 = 950 nM T46685 CA96VH 118731172 IC50 = 100 nM T46685 CSQW02 118988439 IC50 = 41 nM T46685 CH3EG4 118988440 IC50 = 190 nM T46685 CVBF01 127030212 IC50 > 10000 nM T46685 CI93ZA 127030213 IC50 > 10000 nM T46685 C8LQV4 127030516 IC50 = 170 nM T46685 CS12RU 127031435 IC50 = 100 nM T46685 CZXP62 127031750 IC50 = 3900 nM T46685 C3E5YO 127032014 IC50 > 10000 nM T46685 C2ZD8S 127032024 IC50 = 20 nM T46685 CXWY73 127032324 IC50 > 10000 nM T46685 C14RSD 127048474 IC50 = 69 nM T46685 C2LWZ1 129318964 IC50 = 2 nM T46685 C4W6AD 129897084 IC50 = 6.9 nM T46685 C4Z5MQ 131839619 IC50 = 50 nM T46685 C3LR4A 134130122 IC50 > 10000 nM T46685 CAW7I8 134130909 IC50 = 2100 nM T46685 CW84QM 134131222 IC50 > 10000 nM T46685 C6B0RL 134131311 IC50 = 1100 nM T46685 CNJ15A 134132649 IC50 > 10000 nM T46685 C7D9WS 134132677 IC50 = 700 nM T46685 C1UIL9 134135426 IC50 > 10000 nM T46685 C9EQC4 134136966 IC50 > 10000 nM T46685 C4AXE1 134140955 IC50 = 1700 nM T46685 CXA1S4 134142195 IC50 = 1400 nM T46685 CGC6D7 134143498 IC50 > 10000 nM T46685 CSHZ53 134145427 IC50 = 1400 nM T46685 C13TBI 134149173 IC50 > 10000 nM T46685 CP1BV6 134149357 IC50 = 1000 nM T46685 C3HO1K 134152098 IC50 = 890 nM T46685 CZ65XP 134154248 IC50 > 10000 nM T46685 CE42VG 134156031 IC50 > 10000 nM T46685 C8WIV6 134157974 IC50 > 10000 nM T46685 C4QM9O 134397095 IC50 = 66 nM T46685 CQ1K2W 134397387 IC50 = 18 nM T46685 CR08AO 134397388 IC50 = 19 nM T46685 CIN73J 134397390 IC50 = 56 nM T46685 C6I1YX 134397391 EC50 = 9700 nM T46685 CQ9D1Z 134397392 IC50 = 26 nM T46685 CUX8N5 134397449 EC50 = 12200 nM T46685 CDC39N 134397450 EC50 = 4500 nM T46685 C8RN6W 134397451 EC50 = 11700 nM T46685 CE1HY2 134397452 IC50 = 21 nM T46685 CIR51J 134397453 IC50 = 38 nM T46685 C72KFM 134397463 IC50 = 71 nM T46685 CT16YX 134397502 IC50 = 31 nM T46685 CI45HZ 134397798 EC50 = 26400 nM T46685 C2AN7T 134611886 IC50 > 100000 nM T46685 CR1E5Y 135335801 IC50 = 19 nM T46685 CGO0L8 135335871 IC50 = 21 nM T46685 CUG3X6 135335915 IC50 = 20 nM T46685 CJ7FM6 135335919 IC50 = 15 nM T46685 CIOM23 135444382 EC50 = 20000 nM T46685 CJBU04 135590713 IC50 > 10000 nM T46685 CN57OS 136236281 IC50 > 10000 nM T46685 CJC89A 136333957 IC50 = 310 nM T46685 CQ15NR 137631839 IC50 = 40 nM T46685 CI43OC 137632412 EC50 = 26000 nM T46685 CIR86B 137632510 IC50 > 1000 nM T46685 C7E1FL 137633791 IC50 = 24 nM T46685 CH4PN9 137633814 EC50 = 9600 nM T46685 C3BZK6 137633859 IC50 = 64 nM T46685 CI73CB 137634638 IC50 = 280 nM T46685 C3DF5N 137635339 IC50 = 107 nM T46685 CQ2I7Y 137635832 IC50 > 10000 nM T46685 C97FAW 137637167 IC50 = 155 nM T46685 CM7N8S 137637724 IC50 = 29 nM T46685 CRV1E4 137638175 EC50 > 1000000 nM T46685 CL1P2D 137639227 IC50 = 81.6 nM T46685 C89JWP 137639612 IC50 = 439 nM T46685 C84RSO 137640193 IC50 = 18 nM T46685 C3CE9O 137641621 IC50 = 36 nM T46685 CRSQ71 137641785 EC50 = 70000 nM T46685 COH24B 137642226 IC50 = 80 nM T46685 CGCF41 137642917 IC50 = 173 nM T46685 CPO60W 137643573 IC50 > 10000 nM T46685 C75MLQ 137643957 EC50 = 44000 nM T46685 CDA2N6 137644922 IC50 = 5 nM T46685 CWM1P5 137645266 IC50 = 189 nM T46685 CDE8O3 137646031 IC50 = 529 nM T46685 CK6S5T 137646758 EC50 > 1000000 nM T46685 CMI2H3 137647526 EC50 = 117000 nM T46685 C7J9VR 137648478 IC50 > 10000 nM T46685 CCNA21 137648707 IC50 = 45 nM T46685 CNW13G 137648784 EC50 = 12000 nM T46685 CGK5P2 137649037 EC50 = 187000 nM T46685 CS69XL 137649171 IC50 = 30 nM T46685 CM50YV 137649413 IC50 = 139 nM T46685 C9IO5F 137649821 EC50 = 35000 nM T46685 CR0L9E 137651705 IC50 = 4985 nM T46685 CB1H3L 137651798 IC50 > 10000 nM T46685 CDX83M 137654129 EC50 = 34000 nM T46685 CTBD05 137654245 IC50 = 30 nM T46685 CX7V6P 137654671 EC50 > 1000000 nM T46685 CQC49I 137654914 IC50 = 430 nM T46685 C7D9PN 137655679 IC50 = 6 nM T46685 CN1DW2 137655950 IC50 = 7 nM T46685 CYQ61R 137656593 IC50 = 20 nM T46685 C9M5WS 137657239 IC50 = 34 nM T46685 C3Y2CR 137657691 EC50 = 85000 nM T46685 CS5T1Y 137657739 IC50 = 84 nM T46685 C0SBY3 137657758 IC50 = 993 nM T46685 CA10CX 137657812 EC50 = 34000 nM T46685 CD73NA 137658280 IC50 = 66 nM T46685 CX4M8T 137658722 EC50 > 1000000 nM T46685 C25TFP 137659318 IC50 > 1000 nM T46685 CAF68S 137659391 IC50 > 10000 nM T46685 C0U2ZV 137659586 IC50 = 186 nM T46685 CO6H8Z 137660346 EC50 = 8000 nM T46685 CR98AD 137660581 IC50 > 10000 nM T46685 C5J2WV 138728749 IC50 = 786 nM T46685 CVU63L 139582016 IC50 = 1700 nM T46685 C8PH9S 139582017 IC50 = 3100 nM T46685 C6VB3O 145925651 IC50 >= 5000 nM T46685 CX05ZN 145979845 IC50 = 502 nM T46685 CPEC02 145981446 IC50 = 31 nM T46685 CO1S8D 145986658 IC50 = 100 nM T46685 CZU8J6 145992124 IC50 = 270 nM T46685 CK56CB 145993150 IC50 = 730 nM T46685 C2MD1Q 155513187 IC50 > 10000 nM T46685 C86HPW 155518524 IC50 = 13000 nM T46685 CZMF60 155531200 IC50 = 1480 nM T46685 D06CXU 46926513 IC50 = 2 nM T46685 D07OCA 5330812 IC50 = 8.9 nM T46685 D08NQM 5289247 IC50 = 70 nM T46685 D0B5KD 6604931 EC50 = 12000 nM T46685 D0D2FC 2794188 EC50 = 4200 nM T46685 D0D5ZL 369401 IC50 > 10000 nM T46685 D0F5EI 10017019 IC50 = 220 nM T46685 D0O6OH 71553154 IC50 = 1630 nM T46685 D0U3NI 53246941 IC50 = 512 nM T46685 D0UI7U 46926514 IC50 = 68 nM T86014 D07CAQ 3058739 Ki = 3000 nM T86014 D0L0YG 5280335 IC50 = 3860 nM T86014 D0X6BX 15604015 IC50 > 100000 nM T86014 D0AR5O 50916701 Ki = 110 nM T86014 D0DG7E 72735621 IC50 = 5300 nM T86014 D0G2TX 46911228 IC50 = 58 nM T86014 D0TR9T 45256914 IC50 = 68 nM T86014 D0VB2X 72735440 IC50 = 16900 nM T86014 D08SUQ 9925886 IC50 = 7100 nM T86014 C3NIO0 282594 IC50 = 2000 nM T86014 C9GF7W 420266 Ki = 27000 nM T86014 CS3X7Z 2936770 IC50 = 61600 nM T86014 C5CF7V 4132571 IC50 = 40520 nM T86014 C50NXC 5342941 Ki = 1330 nM T86014 CLQ2H6 9564003 IC50 = 23070 nM T86014 C8M9ZK 9630678 IC50 = 22020 nM T86014 CSN36K 9660619 IC50 > 100000 nM T86014 CY6G5N 11305122 Ki = 3000 nM T86014 CACS26 11561968 Ki > 10000 nM T86014 CU0E8O 11690457 Ki > 10000 nM T86014 CB0AP2 11705863 Ki > 10000 nM T86014 CVR8W5 15983462 Ki = 3200 nM T86014 CL7AW8 15983581 Ki = 3100 nM T86014 C7YG1N 24759534 IC50 = 32000 nM T86014 CB1W6K 44404910 IC50 = 650 nM T86014 CCP2U0 45254215 IC50 = 5000 nM T86014 C1U7SH 45254217 IC50 = 25 nM T86014 CQB0K4 45254218 IC50 = 720 nM T86014 CG6S8B 45254415 IC50 = 1100 nM T86014 CUH8L6 45254797 IC50 = 3400 nM T86014 C8ADN2 45254987 IC50 = 4300 nM T86014 CZ17FT 45254988 IC50 = 5000 nM T86014 C6LTF1 45255202 IC50 = 740 nM T86014 CG2BX3 45255825 IC50 = 430 nM T86014 C1XM9Y 45256206 IC50 = 2800 nM T86014 C21KSU 45256386 IC50 > 10000 nM T86014 C83KFZ 45256568 IC50 = 1100 nM T86014 CX6TU7 45256739 IC50 = 61 nM T86014 CMRQ49 45256915 IC50 = 86 nM T86014 CCN34K 45256919 IC50 = 430 nM T86014 C9B3HE 45257096 IC50 = 49 nM T86014 C0FL6I 45257097 IC50 = 380 nM T86014 CVAS82 45257098 IC50 = 210 nM T86014 C1D2FX 45257099 IC50 = 2600 nM T86014 CIW7L6 45257100 IC50 = 620 nM T86014 COSU10 45257101 IC50 = 68 nM T86014 C9DY1H 45267000 IC50 = 2250 nM T86014 CXP98A 45267876 IC50 = 2190 nM T86014 CJTQ86 45269612 IC50 = 2780 nM T86014 CAZR51 45270448 IC50 = 500 nM T86014 CU13FG 45271276 IC50 = 3960 nM T86014 C7I1VS 45273014 IC50 = 3980 nM T86014 CZ5OC1 45483181 IC50 = 180 nM T86014 CR9AD0 45483208 IC50 > 10000 nM T86014 C19PCR 45483233 IC50 = 3500 nM T86014 C6M9FT 45483234 IC50 = 62 nM T86014 C67YVA 45483252 IC50 > 10000 nM T86014 C9E7HG 45483253 IC50 > 10000 nM T86014 CGD8K2 45483254 IC50 = 8300 nM T86014 CJH65X 45483265 IC50 = 2100 nM T86014 CD4P3K 45483266 IC50 = 6200 nM T86014 CR4KW3 45483291 IC50 = 2100 nM T86014 CP24GS 45483298 IC50 = 1600 nM T86014 CQ72RP 45483299 IC50 = 1100 nM T86014 CG8E0V 45483318 IC50 = 3200 nM T86014 C9P4WD 45483319 IC50 > 10000 nM T86014 C7DRY8 46197552 Ki = 200 nM T86014 CE4ZN3 46832080 IC50 = 40 nM T86014 CHUV97 46911229 IC50 = 10 nM T86014 CX02LC 49862315 IC50 > 10000 nM T86014 C4BO1F 49862379 IC50 > 10000 nM T86014 C0PXM2 49862380 IC50 = 610 nM T86014 CLP80E 49862381 IC50 = 2200 nM T86014 CCVQ30 49862427 IC50 = 70 nM T86014 CD74HT 49862540 IC50 = 3800 nM T86014 CD73ZX 49862592 IC50 = 48 nM T86014 CRO9Y8 49862593 IC50 = 30 nM T86014 C09BPE 49862594 IC50 = 110 nM T86014 C6O4ZK 49862647 IC50 = 20 nM T86014 CH3XB1 49862648 IC50 = 56 nM T86014 CND81Y 50916531 Ki = 500 nM T86014 C1KOM0 50916532 Ki = 1300 nM T86014 C9F2AP 50916533 Ki = 390 nM T86014 C6QYN7 50916535 Ki = 130 nM T86014 CKOV69 50916699 Ki = 170 nM T86014 CAT7S6 50916700 Ki = 450 nM T86014 CMCP20 50916702 Ki = 800 nM T86014 CH3M9Z 50916703 Ki = 240 nM T86014 C5T4KE 50916705 Ki = 130 nM T86014 CE89OH 50916894 Ki = 99 nM T86014 C42YBJ 50916895 Ki = 75 nM T86014 CACM70 53247920 Ki = 130 nM T86014 CYM29P 53247958 Ki = 6000 nM T86014 CFY8N9 53247960 Ki = 5400 nM T86014 CV37EJ 53247962 Ki = 9000 nM T86014 CT5G7A 53248010 Ki = 2000 nM T86014 C5SOT7 53248014 Ki = 47 nM T86014 CV0ZA9 53248130 Ki = 110 nM T86014 C3Q6KD 53248235 Ki = 5000 nM T86014 CZ5WB2 53248278 Ki = 1500 nM T86014 C5XG8H 53248469 Ki = 1300 nM T86014 CM70XH 53248470 Ki = 95 nM T86014 CL9A3O 53248471 Ki = 4000 nM T86014 CTSN72 53248514 Ki = 1600 nM T86014 CL0D2O 53248519 Ki = 16000 nM T86014 C5DMR6 53494962 IC50 = 820 nM T86014 CT03KQ 56839813 Ki = 60000 nM T86014 CV8X1J 56840034 Ki = 22000 nM T86014 CK5A3Q 56929818 IC50 = 20 nM T86014 CCG07K 57390485 Ki > 100000 nM T86014 C4I5LS 57390557 Ki = 32000 nM T86014 CZ0TU3 57390558 Ki = 40000 nM T86014 CUY42W 57395844 Ki = 22000 nM T86014 C3BJE5 57395846 Ki = 70000 nM T86014 C6YSW2 57399302 Ki > 100000 nM T86014 CXJ63M 59603829 IC50 > 100000 nM T86014 CQEU96 59603842 IC50 > 10000 nM T86014 C1MR8Q 60097495 IC50 > 10000 nM T86014 C4R8BS 60149004 Ki = 40 nM T86014 CUC7B3 66557964 IC50 = 29000 nM T86014 C5DGR9 69036886 IC50 = 10000 nM T86014 CPR8M7 71449578 Ki = 15000 nM T86014 CH5YO1 71451384 Ki = 35000 nM T86014 C4V8NY 71453197 Ki = 35000 nM T86014 CEC75Q 71458557 Ki = 36000 nM T86014 CH19YZ 71460405 Ki = 13000 nM T86014 CZEM14 71462095 Ki = 27000 nM T86014 C91MOC 71521167 Ki = 200 nM T86014 CS92CX 71546264 IC50 = 3600 nM T86014 C19SBT 71602841 EC50 = 5700 nM T86014 C7EAG6 71602883 EC50 = 8300 nM T86014 CQ7R2F 71627420 IC50 = 20 nM T86014 CA6MN7 71661218 Ki = 1000 nM T86014 C58SXV 71714682 IC50 > 10000 nM T86014 C41HDP 71727564 Ki > 10000 nM T86014 C2JVX0 71727565 Ki > 10000 nM T86014 C6DSB9 71727676 Ki > 10000 nM T86014 CHB2G5 71727800 Ki = 48 nM T86014 C7HM8J 71812415 IC50 = 3 nM T86014 CQOM26 71812416 IC50 = 5 nM T86014 CIHY54 71812417 IC50 = 4 nM T86014 C1XR2P 71812418 IC50 = 3 nM T86014 CD51FM 71813340 IC50 = 1600 nM T86014 C23DVM 71813341 IC50 = 990 nM T86014 C4BJU1 71813342 IC50 = 580 nM T86014 CH75OI 71813505 IC50 = 2300 nM T86014 C0Q7AR 71813506 IC50 = 140 nM T86014 CO4E5N 71813507 IC50 = 920 nM T86014 CD5B1M 71813508 IC50 = 2100 nM T86014 CC4MZ3 71813509 IC50 = 1800 nM T86014 CD8G2B 71813510 IC50 > 10000 nM T86014 CNF79K 71813670 IC50 = 1000 nM T86014 C42RXL 71813671 IC50 = 3100 nM T86014 C2YP9U 71813673 IC50 = 80 nM T86014 CC0Z9Y 71813674 IC50 = 1100 nM T86014 CR20UF 71813675 IC50 = 20 nM T86014 CZ4N6I 71813828 IC50 = 220 nM T86014 CDG82F 71813829 IC50 = 450 nM T86014 CA29MU 71813830 IC50 = 230 nM T86014 CHB8F6 71813831 IC50 = 2500 nM T86014 C8GX0A 71813832 IC50 = 130 nM T86014 CS3U7T 71813975 IC50 = 30 nM T86014 C3WXA8 71813976 IC50 = 410 nM T86014 C6JX4K 71813977 IC50 = 30 nM T86014 C2VB7R 71814309 IC50 = 2000 nM T86014 CNU3R2 71814310 IC50 = 120 nM T86014 CGI8O9 71814493 IC50 = 150 nM T86014 CGCK24 71814494 IC50 = 1100 nM T86014 CQ3JF6 71814495 IC50 = 2100 nM T86014 CZNC03 71814496 IC50 = 170 nM T86014 C8V1TU 71814497 IC50 = 270 nM T86014 CZVX43 71814498 IC50 = 80 nM T86014 CC43NW 71814674 IC50 > 10000 nM T86014 C1ZNP6 71814675 EC50 = 310 nM T86014 C3Y6GW 71814676 EC50 = 130 nM T86014 CND38P 71814677 EC50 = 80 nM T86014 C4HE3B 71814678 IC50 = 320 nM T86014 C3HR1T 71814679 IC50 = 20 nM T86014 C6P8KM 71814846 IC50 = 10 nM T86014 C9BJZ6 71814847 EC50 = 870 nM T86014 CQ62UK 71814848 EC50 = 120 nM T86014 C9FK2A 71814849 EC50 = 1200 nM T86014 CEP2B5 71814850 IC50 = 8 nM T86014 CW1X0Y 71814851 IC50 = 7 nM T86014 CRM17W 71815023 IC50 = 30 nM T86014 C6KC3P 71815024 EC50 = 370 nM T86014 C8RPW2 71815025 IC50 > 5000 nM T86014 CA68ON 71815026 IC50 = 5 nM T86014 CR8Z6C 71815027 EC50 = 280 nM T86014 CHY3O8 71815028 EC50 = 850 nM T86014 CBXD42 72735619 IC50 = 2200 nM T86014 CB24ZV 73265274 Ki = 4.3 nM T86014 C3A4KF 73349099 IC50 = 6100 nM T86014 CE7UR8 73353633 Ki = 10000 nM T86014 CF83GY 76325790 IC50 = 69000 nM T86014 C5FDA8 76329372 IC50 = 27800 nM T86014 C1HW4B 89735655 IC50 > 100000 nM T86014 CIW6T4 89740017 Ki = 400 nM T86014 C9FM2Y 89740586 Ki = 1600 nM T86014 CFH3S4 89740671 Ki = 40 nM T86014 CC6MX1 89741221 Ki = 3000 nM T86014 C8ON1V 89741310 Ki = 260 nM T86014 CCWB78 89741619 Ki > 10000 nM T86014 CBR42S 101913779 IC50 = 7300 nM T86014 C93YFS 118255060 Ki = 440 nM T86014 CE24JK 118255132 Ki = 13000 nM T86014 C48KEV 118611394 IC50 > 20000 nM T86014 CLQ9R7 118611411 IC50 = 3100 nM T86014 C9Q0DC 118734327 IC50 = 58 nM T86014 CN9P8D 118734390 Ki = 13000 nM T86014 CCTD29 122365196 IC50 > 30000 nM T86014 CK16NT 122365197 IC50 = 220 nM T86014 CFD9T6 122365198 IC50 = 4000 nM T86014 C5PH3C 127027128 IC50 = 20 nM T86014 C0EQ9W 127043058 Ki = 980 nM T86014 CBI8C4 127045038 Ki = 4600 nM T86014 C7JF3L 127045539 Ki = 2500 nM T86014 C54NZV 127045540 Ki = 100 nM T86014 C5V8PK 127045541 Ki = 70 nM T86014 C1EJN8 127048670 IC50 = 63240 nM T86014 CR5J7D 127048671 IC50 = 52100 nM T86014 CI6VY1 127048672 IC50 = 45790 nM T86014 C3T2NZ 127048673 IC50 = 19570 nM T86014 CIOB05 127049002 IC50 > 100000 nM T86014 C51ZEV 127049003 IC50 = 16260 nM T86014 CCH2S3 127049291 IC50 = 32730 nM T86014 C72VGW 127049294 IC50 = 69440 nM T86014 CV1M5H 127049332 IC50 = 40550 nM T86014 CP5TM3 127049333 IC50 = 20610 nM T86014 C32ETI 127049334 IC50 = 18440 nM T86014 C9VJX7 127049335 IC50 = 4360 nM T86014 C0PNK3 127049336 IC50 > 100000 nM T86014 C2MHI6 127049994 IC50 > 100000 nM T86014 CJ51CK 127050232 Ki > 20000 nM T86014 CNV12K 127050290 IC50 > 100000 nM T86014 CJT87U 127050865 IC50 > 100000 nM T86014 CY6MD3 127050920 IC50 = 15010 nM T86014 CI9E4G 127050921 IC50 = 54720 nM T86014 CRCG86 127050922 IC50 = 37400 nM T86014 CO0M4W 127050923 IC50 > 100000 nM T86014 CVIN74 127050924 IC50 = 45760 nM T86014 CMB5C6 127051152 Ki = 730 nM T86014 C0NXA4 127051153 Ki = 930 nM T86014 CTSP67 127051186 IC50 = 27740 nM T86014 CJ3KN5 127051492 IC50 > 100000 nM T86014 CD4P9L 127051493 IC50 > 100000 nM T86014 C8JW6R 127051494 IC50 = 15530 nM T86014 CD5FY0 127051495 IC50 > 100000 nM T86014 C5C2UN 127051496 IC50 > 100000 nM T86014 CP9O2Q 127051497 IC50 = 16480 nM T86014 C4U3VW 127051810 IC50 = 45380 nM T86014 CDV4I7 127052117 IC50 = 85260 nM T86014 C5W3BG 127052118 IC50 = 31300 nM T86014 C3W2BY 127052119 IC50 = 20520 nM T86014 C6B5ML 127052120 IC50 = 8570 nM T86014 CKB92N 127052121 IC50 > 100000 nM T86014 CFZ6M0 127052140 Ki = 7200 nM T86014 CFQ63S 127052141 Ki > 10000 nM T86014 C1XRW2 127052719 IC50 > 100000 nM T86014 CZY17D 127052720 IC50 > 100000 nM T86014 CB6JF5 127052721 IC50 > 100000 nM T86014 CV0LF4 127052728 IC50 > 100000 nM T86014 C63CWH 127052729 IC50 = 5000 nM T86014 C7BMU9 127052730 IC50 > 100000 nM T86014 CL02DX 127052731 IC50 > 100000 nM T86014 CH8PE9 127052732 IC50 > 100000 nM T86014 CG4KH8 127052733 IC50 = 25320 nM T86014 CZWF94 127052734 IC50 > 100000 nM T86014 C58VJN 127053007 IC50 = 36800 nM T86014 CCJ71P 127053008 IC50 > 100000 nM T86014 C0U1SE 127053009 IC50 > 100000 nM T86014 CW3EN2 127053010 IC50 = 35220 nM T86014 C54FXD 134957362 IC50 > 10000 nM T86014 C1R5NL 135515522 Ki = 1060 nM T86014 C0YDR9 137553159 IC50 = 1200 nM T86014 CJHA89 137631941 IC50 = 4600 nM T86014 CG46PI 137632626 IC50 = 0.03 nM T86014 C4FMC0 137632632 IC50 = 290 nM T86014 CYB4Z5 137633994 IC50 = 710 nM T86014 CF8T9O 137634221 IC50 = 1.7 nM T86014 CAW7X5 137634618 IC50 = 1 nM T86014 CV65UW 137634788 IC50 = 0.17 nM T86014 CPJN61 137635064 Ki = 300 nM T86014 CM9X6B 137635845 IC50 = 880 nM T86014 CU65BI 137636078 IC50 > 100000 nM T86014 CX8DI3 137636195 IC50 = 16000 nM T86014 CC30PZ 137638678 Ki = 700 nM T86014 C2ZEL8 137639097 IC50 > 30000 nM T86014 CB3D4T 137641685 IC50 > 30000 nM T86014 C9FID2 137642040 IC50 > 30000 nM T86014 C8AMX6 137642427 IC50 = 4 nM T86014 C1T8DM 137642521 IC50 = 9800 nM T86014 CSQH31 137643140 IC50 = 4.8 nM T86014 C9W3NK 137643775 IC50 = 0.3 nM T86014 CDH76B 137644043 IC50 = 12000 nM T86014 COMC94 137646013 Ki = 800 nM T86014 CAME30 137646035 IC50 = 870 nM T86014 C51LSX 137647661 IC50 = 420 nM T86014 CQLJ28 137649154 IC50 > 30000 nM T86014 C92CZT 137649534 IC50 = 28 nM T86014 C3KN9J 137649735 IC50 = 380 nM T86014 CDT06A 137649743 Ki = 120 nM T86014 CP63XR 137650218 Ki = 820 nM T86014 CQ2M6U 137650955 IC50 = 2.6 nM T86014 C7QT3K 137651095 Ki = 730 nM T86014 C9KMW8 137651971 IC50 = 1100 nM T86014 CF0Q3L 137652248 Ki = 9000 nM T86014 CA84YU 137653104 IC50 = 2800 nM T86014 CTWO43 137653344 Ki = 12000 nM T86014 CABF71 137653763 Ki = 5000 nM T86014 CXPR04 137653767 IC50 = 250 nM T86014 CUB26L 137653999 IC50 = 439 nM T86014 C8J0QG 137655784 IC50 = 4 nM T86014 C7I1HX 137657086 IC50 = 10 nM T86014 CLF8M0 137657883 IC50 = 1.7 nM T86014 CKH03X 137657977 IC50 = 3.5 nM T86014 CX63PI 137658079 IC50 = 9600 nM T86014 CHUZ37 137658235 IC50 > 30000 nM T86014 C8P7TG 137659208 IC50 = 3100 nM T86014 CFBW57 137660541 IC50 > 100000 nM T86014 CA09GJ 137660569 IC50 = 27000 nM T86014 CH2AN7 137660780 IC50 = 180 nM T86014 CKOQ53 137660812 IC50 = 670 nM T86014 CK7LE0 137661361 IC50 = 1400 nM T86014 C2DFC3 145950249 IC50 = 12000 nM T86014 C9HR3A 145952277 IC50 = 60000 nM T86014 CZC40Q 145959201 IC50 = 55000 nM T86014 CK3D2P 154699447 IC50 = 14 nM T86014 C0QY4W 154699448 IC50 = 4130 nM T86014 C8NI1W 154699449 IC50 = 765 nM T86014 CYUT01 154699450 IC50 = 2360 nM T86014 C1CAT9 155517174 IC50 = 11 nM T86014 CNB93E 155519701 IC50 > 3000 nM T86014 CSGJ75 155523497 IC50 = 39 nM T86014 C89YXV 155524292 EC50 > 950 nM T86014 CF78NS 155524444 EC50 > 800 nM T86014 CTP85C 155525319 IC50 = 170 nM T86014 CZ82OI 155525383 IC50 = 44 nM T86014 CXB1Q7 155528975 EC50 > 800 nM T86014 CON56I 155531486 EC50 > 1000 nM T86014 C0MC9O 155535418 IC50 = 26 nM T86014 C31DCI 155536233 EC50 > 1000 nM T86014 CC62JR 155536715 IC50 = 9 nM T86014 C0ITD5 155555664 IC50 = 41 nM T86014 CR96ED 155557208 IC50 > 3000 nM T86014 CZ06PJ 155564368 EC50 > 500 nM T86014 CQL4F1 155564588 IC50 = 137 nM T86014 CC9F8Z 155569662 EC50 > 550 nM T86014 D00YNY 753704 Ki = 500 nM T86014 D01UUZ 45254608 IC50 = 2200 nM T86014 D01XSX 45256207 IC50 = 4000 nM T86014 D05SLY 44815217 Ki = 10000 nM T86014 D08SND 66577038 IC50 = 2 nM T86014 D0E3LA 45255203 IC50 = 5000 nM T86014 D0H2LN 71458556 IC50 > 50000 nM T86014 D0M9DT 5282309 Ki = 5000 nM T86014 D0P5TI 58441401 IC50 > 1000 nM T86014 D0TC4I 45483175 IC50 = 50 nM T20958 D09AVU 46202376 IC50 = 82 nM T20958 D0AT0A 46208464 IC50 = 18 nM T20958 D0I0BN 11177829 IC50 = 1.995 nM T20958 D0I8ZE 49862986 IC50 = 7 nM T20958 D0M3DM 8088007 IC50 = 27 nM T20958 D0WI0P 44156964 IC50 = 1.2 nM T20958 C2VFW6 3989078 IC50 = 2800 nM T20958 CTI78W 16196125 IC50 = 51 nM T20958 C49QTJ 35277770 IC50 = 794.33 nM T20958 C0PO5V 44123843 EC50 = 0.6761 nM T20958 CK3V8D 44634514 IC50 = 35000 nM T20958 CH9FE5 44634521 IC50 = 27000 nM T20958 C9DYV0 44634539 IC50 = 7300 nM T20958 CPU06K 44634544 IC50 = 4030 nM T20958 CG8W3D 44634570 IC50 = 1000 nM T20958 C9R6NO 46189900 IC50 = 387 nM T20958 CT64KQ 46202039 IC50 = 114 nM T20958 C9ZUE4 46202040 IC50 = 145 nM T20958 CX6G3V 46202041 IC50 = 851 nM T20958 C6SZ5E 46202042 IC50 = 2179 nM T20958 C25GBV 46205607 IC50 = 321 nM T20958 C7HKW6 46205608 IC50 = 254 nM T20958 CE82RV 46206598 IC50 = 46 nM T20958 CY89ER 46206599 IC50 = 380 nM T20958 CH3RQ6 46206931 IC50 = 369 nM T20958 CL2NS3 46206933 IC50 = 351 nM T20958 CK6V4Y 46206934 IC50 = 1325 nM T20958 CCSB86 46930969 IC50 = 0.96 nM T20958 CFW9U8 46930970 IC50 = 2100 nM T20958 CZ9EN2 46930971 IC50 < 0.5 nM T20958 CHA32Z 46930978 IC50 = 13 nM T20958 C04JWM 49862947 IC50 = 1577 nM T20958 CTL49W 49862948 IC50 = 725 nM T20958 CE18GJ 49862983 IC50 = 326 nM T20958 C4OVU9 49862984 IC50 = 31 nM T20958 CFIQ68 49862985 IC50 = 144 nM T20958 C6IRJ1 49863016 IC50 = 14 nM T20958 CJ2XV0 49863017 IC50 = 22 nM T20958 CAPG01 49863070 IC50 = 103 nM T20958 C60HJV 49863071 IC50 = 398 nM T20958 CMG9L5 50925456 IC50 = 19.95 nM T20958 CMF7T6 50925457 IC50 = 10 nM T20958 CGLX34 52942376 IC50 > 5011.87 nM T20958 CP3C4V 52942771 IC50 = 31.62 nM T20958 C5ZS3A 52944769 IC50 = 251.19 nM T20958 C5KPW2 52945990 IC50 > 5011.87 nM T20958 CG4IB9 52948466 IC50 > 5011.87 nM T20958 C39YQE 56659483 IC50 = 154 nM T20958 CNK0C5 56659484 IC50 = 358 nM T20958 C4V9SR 56659485 IC50 = 134 nM T20958 CPOX85 56659486 IC50 = 96 nM T20958 CL6D1E 56662909 IC50 = 50 nM T20958 CR6S4G 56662945 IC50 = 92 nM T20958 CV76LA 56662946 IC50 = 90 nM T20958 CM2P9C 56666418 IC50 = 3166 nM T20958 CYV3Q9 56666419 IC50 = 239 nM T20958 CNY09J 56669801 IC50 = 1458 nM T20958 C79EQU 56669836 IC50 = 1500 nM T20958 CU97VE 56676652 IC50 = 92 nM T20958 CD6WC8 56676659 IC50 = 336 nM T20958 C4M0IY 56676660 IC50 = 635 nM T20958 C3MBQ9 56676661 IC50 = 131 nM T20958 CD39KX 56676662 IC50 = 126 nM T20958 C71RVE 56679926 IC50 = 660 nM T20958 CM3EX8 56679981 IC50 = 1725 nM T20958 C4JOH7 56683317 IC50 = 138 nM T20958 CR05ML 56683318 IC50 = 95 nM T20958 CR89TK 72735786 IC50 = 2500 nM T20958 CUO0D9 72735787 IC50 = 1300 nM T20958 CP79TV 72735979 IC50 = 2100 nM T20958 CYLO49 72735981 IC50 < 0.5 nM T20958 CQCI69 72736185 IC50 = 3.2 nM T20958 C5LO9T 72736186 IC50 = 3.4 nM T20958 C40PKO 72736187 IC50 = 9.2 nM T20958 CP1L3G 72736188 IC50 = 2.2 nM T20958 CL95CX 72736369 IC50 = 400 nM T20958 C69KEZ 72736370 IC50 = 170 nM T20958 C7TNG1 72736371 IC50 = 23 nM T20958 CF31HN 72736372 IC50 = 45 nM T20958 CTA37O 72736542 IC50 = 64 nM T20958 C8Z6IP 72736543 IC50 = 71 nM T20958 CW2J8V 72736544 IC50 = 9 nM T20958 CB4L5O 76320765 IC50 = 4900 nM T20958 CGP4Z6 155544367 IC50 = 3900 nM T20958 CADQ93 155557362 IC50 = 5770 nM T20958 D03EJP 11374217 IC50 = 48 nM T20958 D09RIC 46203026 IC50 = 43 nM T53811 D0K8KX 5280343 IC50 > 20000 nM T53811 D0G3TK 5280863 IC50 > 20000 nM T53811 D0NJ4H 5281670 IC50 = 4000 nM T53811 D0T3PW 5281672 IC50 = 850 nM T99816 C60UTZ 6324606 EC50 = 41 nM T99816 C8E4SI 11766466 Ki = 0.7 nM T99816 CF0G4N 16201612 Ki = 0.15 nM T99816 CPDR90 21255267 Ki = 1500 nM T99816 CX26WC 21255272 Ki > 10000 nM T99816 CQ6X4A 21255273 Ki > 10000 nM T99816 CPB38K 21255275 Ki > 10000 nM T99816 CXR36V 21255282 Ki > 10000 nM T99816 CNW89T 25026445 IC50 > 10000 nM T99816 CND1W8 44300286 EC50 = 84 nM T99816 C3UL9V 44321006 Ki = 3.7 nM T99816 C6B3CL 44321034 Ki = 37 nM T99816 CVR13I 44321035 Ki = 1254 nM T99816 C0F3LI 44321036 Ki = 404 nM T99816 CVGO97 44321037 Ki = 124 nM T99816 C1RQG9 44321039 Ki = 9 nM T99816 C86MBK 44321083 Ki = 85 nM T99816 CB31KF 44321084 Ki = 149 nM T99816 C5CKH1 44321085 Ki = 1096 nM T99816 C43NHF 44321117 Ki = 35 nM T99816 CKSE24 44321157 Ki = 273 nM T99816 C3WRP8 44321158 Ki = 32 nM T99816 CZ6RU8 44321211 Ki = 89 nM T99816 C6VML9 44321212 Ki = 6.4 nM T99816 CE1W0A 44321244 Ki = 33 nM T99816 CFGW75 44321245 Ki = 5.8 nM T99816 CTDB98 44321246 Ki = 85 nM T99816 C4XF2V 44322126 Ki > 10000 nM T99816 CP50SE 44322138 Ki = 0.7 nM T99816 C52NMY 44322245 Ki > 10000 nM T99816 CJZ18R 44322247 Ki > 10000 nM T99816 C0H7ZD 44322273 Ki > 10000 nM T99816 C1X9YD 44322303 Ki > 10000 nM T99816 C9YD7L 44322304 Ki > 10000 nM T99816 C4NBE8 44322341 Ki > 10000 nM T99816 CFB2U7 44322391 Ki > 10000 nM T99816 C83QYU 44322460 Ki > 10000 nM T99816 C9B4ZC 44322461 Ki > 10000 nM T99816 CRS04C 44388192 IC50 = 0.72 nM T99816 CFWA84 44454030 EC50 = 0.373 nM T99816 C7SW1I 44589983 EC50 = 0.06 nM T99816 C2G4YW 46882011 IC50 > 10000 nM T99816 C7ANC0 57391433 Ki > 10000 nM T99816 COU60J 57402754 Ki > 10000 nM T99816 C4INR9 57568258 IC50 = 22.9 nM T99816 CWMQ18 72704870 IC50 = 8.3 nM T99816 C72STJ 72705066 IC50 = 23 nM T99816 CJC7E2 73345589 IC50 = 0.47 nM T99816 CPC49J 73345664 IC50 = 1.45 nM T99816 CO84AR 73350855 IC50 = 5.3 nM T99816 C5X1KD 73351696 IC50 = 1.94 nM T99816 CIV74J 73353243 IC50 = 0.59 nM T99816 CS6Z5R 73356238 IC50 = 0.85 nM T99816 CLZ7J2 90663965 EC50 = 12200 nM T99816 CC5J7U 90663970 EC50 = 19100 nM T99816 CU3SH6 118728504 Ki = 0.5 nM T99816 D02TPY 25025860 IC50 = 6400 nM T99816 D03TEJ 5311352 Ki > 10000 nM T99816 D07IAK 9937534 Ki = 17 nM T99816 D0I5CS 9829828 Ki = 1 nM T99816 D0MH6P 11434815 IC50 = 1.3 nM T99816 D0R8TG 11389266 IC50 = 0.08 nM T20585 CCAN47 9801356 IC50 = 6.5 nM T20585 C6DP4S 10003041 IC50 = 8.2 nM T20585 C09RKT 10071438 IC50 = 61 nM T20585 CHP24I 10071935 IC50 = 2.2 nM T20585 C63CAY 10321901 IC50 = 0.7 nM T20585 C4DXB7 10340781 IC50 = 21 nM T20585 C6LUZ0 23071543 IC50 = 5200 nM T20585 CF7M4B 23071563 IC50 = 7 nM T20585 C68KRW 23071571 IC50 = 310 nM T20585 C9RQD8 44208030 IC50 = 1.9 nM T20585 CF9IN6 44422639 IC50 = 190 nM T20585 CLW5S1 44422642 IC50 = 170 nM T20585 C4VW6N 44422645 IC50 = 380 nM T20585 CP8FN2 44422650 IC50 = 3000 nM T20585 C3UP4Y 44422652 IC50 = 1100 nM T20585 C5MS8J 44422655 IC50 = 130 nM T20585 CY2W9R 44422656 IC50 = 660 nM T20585 CFS8O6 44422657 IC50 = 8200 nM T20585 CS50TP 44422658 IC50 = 410 nM T20585 CVF68I 44422659 IC50 = 64 nM T20585 CLH62W 44422660 IC50 = 100 nM T20585 CHGB27 44422661 IC50 = 88 nM T20585 CAG5D6 44422662 IC50 = 45 nM T20585 CQK4J1 44422663 IC50 = 30 nM T20585 C98AFC 44422664 IC50 = 83 nM T20585 CS3HU2 44561016 IC50 = 2000 nM T20585 CRM68E 44561017 IC50 = 36 nM T20585 CFN56B 44561018 IC50 = 130 nM T20585 CH8GM0 44561019 IC50 = 25 nM T20585 C26KXE 44561062 IC50 = 19 nM T20585 C6FVT1 44561128 IC50 = 2.1 nM T20585 CS13DE 44561129 IC50 = 310 nM T20585 CWQ0D2 44561130 IC50 = 1.6 nM T20585 C60ZKU 44561161 IC50 = 5.5 nM T20585 CR35PN 44561162 IC50 = 1.8 nM T20585 C75ZKA 44561163 IC50 = 0.7 nM T20585 CD4U5Z 44561164 IC50 = 88 nM T20585 CWE4G2 44561384 IC50 = 95 nM T20585 C0E5YW 44561385 IC50 = 81 nM T20585 C6GT8V 44561427 IC50 = 98 nM T20585 CG0SJ6 44561428 IC50 = 16 nM T20585 CX42EU 44561429 IC50 = 650 nM T20585 CCFE41 44561430 IC50 = 120 nM T20585 CA2N0M 44561473 IC50 = 6.2 nM T20585 C9Z6EB 44561474 IC50 = 17 nM T20585 CW72PY 44561514 IC50 = 1.4 nM T20585 CKC1P0 44561515 IC50 = 1.8 nM T20585 C12CMX 44561516 IC50 = 650 nM T20585 C41YZC 44561517 IC50 = 11 nM T20585 CDU4R8 44561553 IC50 = 22 nM T20585 CMG8U1 44561554 IC50 = 7.9 nM T20585 C8X1YW 44561555 IC50 = 25 nM T20585 CSKD78 44561582 IC50 = 38 nM T20585 C96KRO 44561583 IC50 = 23 nM T20585 CDAB83 46227231 IC50 = 4.7 nM T20585 CXF75A 46227232 IC50 = 4100 nM T20585 CANR40 46227235 IC50 = 400 nM T20585 CS21GL 46227244 IC50 = 220 nM T20585 C9C5QE 46227245 IC50 = 120 nM T20585 C05VWA 46227254 IC50 = 37 nM T20585 C5VUH7 46227255 IC50 = 12 nM T20585 C5W7JV 46227259 IC50 = 3.2 nM T20585 C8E0HG 46227260 IC50 = 5.6 nM T20585 CRZS59 46227265 IC50 = 34 nM T20585 CM31OQ 46227277 IC50 = 26 nM T20585 CFYN81 46227332 IC50 = 8300 nM T20585 C9G1AS 56950508 IC50 = 2700 nM T20585 C8U3VT 59902815 IC50 = 120 nM T20585 CE85MZ 71450426 IC50 = 3200 nM T20585 C0YMF6 86292327 IC50 = 44 nM T20585 C5KUD6 86292328 IC50 = 28 nM T20585 CI9XT2 86292329 IC50 = 89 nM T20585 COP60F 86292515 IC50 = 120 nM T20585 CV0AW7 86292516 IC50 = 270 nM T20585 CE93RU 86292517 IC50 = 230 nM T20585 CAG5Z3 86292518 IC50 = 120 nM T20585 C25UFB 86292519 IC50 = 380 nM T20585 C1AO2V 127037984 IC50 = 2400 nM T20585 CC0YS1 127039143 IC50 = 140 nM T20585 C9B2UK 127039144 IC50 = 870 nM T20585 C5YP4F 127039145 IC50 = 1250 nM T20585 C58MXN 127039152 IC50 = 340 nM T20585 C09JTZ 127039397 IC50 = 540 nM T20585 C7J3HZ 127039398 IC50 = 1070 nM T20585 COL74J 127039711 IC50 = 1800 nM T20585 CZG8Q1 127039722 IC50 = 410 nM T20585 CU4MA7 127039723 IC50 = 270 nM T20585 C79QOU 127041711 IC50 = 480 nM T20585 CU4I6P 127041752 IC50 = 4500 nM T20585 CZX34A 127041753 IC50 = 4200 nM T20585 CQB07Y 127042069 IC50 = 6100 nM T20585 CM6F2Q 127042070 IC50 = 5200 nM T20585 C8HG0P 127042071 IC50 = 4000 nM T20585 CV5ML8 127042072 IC50 = 5200 nM T20585 CJPG12 127042074 IC50 = 14900 nM T20585 C5N9CI 127042075 IC50 = 8100 nM T20585 CI9JR7 127042076 IC50 = 4100 nM T20585 C61QNZ 127042077 IC50 = 3500 nM T20585 C8MPC4 127042080 IC50 = 6600 nM T20585 CK3J8Z 127042081 IC50 = 8600 nM T20585 CZU57E 127042082 IC50 = 3700 nM T20585 CI6XR7 127042326 IC50 = 250 nM T20585 CC1EI4 127042327 IC50 = 740 nM T20585 C4H6CX 127042328 IC50 = 3430 nM T20585 C6ZHL7 127042429 IC50 = 89600 nM T84726 D03KKR 3547 IC50 = 180 nM T84726 C9KT7Q 163751 IC50 = 180 nM T84726 CGN6T0 9835432 IC50 = 70 nM T84726 C9C8EY 9836178 IC50 = 240 nM T84726 CHP4O1 9840006 IC50 = 25 nM T84726 C5XMP4 9857714 IC50 = 20 nM T84726 C56GPV 9858433 IC50 = 25 nM T84726 C0T6NW 9900683 IC50 = 32 nM T84726 CC1J0A 9900997 IC50 = 85 nM T84726 C1SKR3 9965608 IC50 = 180 nM T84726 CY89AV 9967878 IC50 = 10 nM T84726 CA74YF 9974356 IC50 = 65 nM T84726 CO36BZ 10020867 IC50 = 210 nM T84726 C1X6HO 10041590 IC50 = 205 nM T84726 CQ7N3R 10064487 IC50 = 235 nM T84726 CMSQ48 10065796 IC50 = 75 nM T84726 C3H4ST 10245340 IC50 = 310 nM T84726 C2QM0N 10315045 IC50 = 100 nM T84726 C62PXQ 10360623 IC50 = 185 nM T84726 CZ65IG 10427217 IC50 = 65 nM T84726 C6BM8O 10428037 IC50 = 265 nM T84726 C9NZT2 10471319 IC50 = 95 nM T84726 CR92GA 11537005 IC50 = 75 nM T84726 CZR39O 11723420 IC50 = 275 nM T84726 CW53JC 11998038 Ki = 6 nM T84726 COTM04 17838031 IC50 = 345 nM T84726 CLR83G 17838080 IC50 = 210 nM T84726 CMEZ85 17838131 IC50 = 220 nM T84726 C30WCJ 17838150 IC50 = 270 nM T84726 C0Z6LA 17838157 IC50 = 340 nM T84726 CGFW16 17838175 IC50 = 20 nM T84726 CZT35Q 17838190 IC50 = 260 nM T84726 CKF51W 17838202 IC50 = 440 nM T84726 CGWH21 17838205 IC50 = 320 nM T84726 CU4F9X 17838266 IC50 = 780 nM T84726 CCR8J4 17838276 IC50 > 10000 nM T84726 C6K9RC 21098468 IC50 = 13 nM T84726 CMF27K 21098469 IC50 = 45 nM T84726 C7WBX4 21098475 IC50 = 80 nM T84726 CFB3T6 21098478 IC50 = 19 nM T84726 C1B7UA 21098479 IC50 = 290 nM T84726 C9T8FA 21098480 IC50 = 20 nM T84726 CMA42E 21098488 IC50 = 11 nM T84726 CDU6P0 21098489 IC50 = 290 nM T84726 C9JI3T 21098490 IC50 = 24 nM T84726 CK51MC 21098512 IC50 = 3 nM T84726 CN8F1W 21098519 IC50 = 16 nM T84726 CW0BP6 21098523 IC50 = 9 nM T84726 C1WM8S 21098530 IC50 = 87 nM T84726 CXQ49I 22933424 IC50 = 136 nM T84726 C5XB1S 22933917 IC50 = 540 nM T84726 CZWI08 25093233 IC50 = 1.5 nM T84726 C92QDU 42611189 Ki = 210 nM T84726 CAO2T4 42634832 Ki = 560 nM T84726 CN79ZK 44421854 IC50 = 240 nM T84726 C9OBD5 44421855 IC50 = 72 nM T84726 CFKZ21 44421856 IC50 = 190 nM T84726 C7N8YR 44421860 IC50 = 11 nM T84726 C5HCK8 44421861 IC50 > 1000 nM T84726 CQW39E 44421862 IC50 = 5 nM T84726 CQ07XN 44421867 IC50 = 3 nM T84726 C7SL3R 44421868 IC50 = 65 nM T84726 CJ2XH8 44421869 IC50 = 180 nM T84726 C7L2UB 44421888 IC50 = 100 nM T84726 CUD80R 44421889 IC50 = 10 nM T84726 C65LTK 44421899 IC50 = 150 nM T84726 CV5IJ4 44421900 IC50 > 10000 nM T84726 C5W0IT 44421911 IC50 = 7900 nM T84726 C6VX5S 44421912 IC50 > 10000 nM T84726 C3K7NQ 44421913 IC50 = 18 nM T84726 CEQ1G8 44421916 IC50 > 10000 nM T84726 C7PCB4 44421917 IC50 = 85 nM T84726 C5T6WC 44421922 IC50 = 35 nM T84726 C87DBT 44421923 IC50 = 10 nM T84726 CU0Q2T 44422390 IC50 = 140 nM T84726 CP12FE 44422393 IC50 = 440 nM T84726 CX6PZ9 51003130 IC50 = 12 nM T84726 C5JYB8 68515257 IC50 = 116 nM T84726 CL8SO7 68516150 IC50 = 49800 nM T84726 CHT6K9 118728811 Ki > 4000 nM T84726 CUA3Y2 118728812 Ki > 4000 nM T84726 CDQ78G 118728813 Ki = 250 nM T84726 CZ6XL7 118728814 Ki > 4000 nM T84726 CMO67K 118728815 Ki > 4000 nM T84726 CR2M0Q 118728816 Ki > 4000 nM T84726 C62SCL 118728817 Ki > 4000 nM T84726 CSB30C 118728819 Ki = 980 nM T84726 CV7XU8 118728820 Ki = 1500 nM T84726 C3J1EX 118728821 Ki > 4000 nM T84726 CIWB78 118728822 Ki > 4000 nM T84726 CP18SE 118728823 Ki = 310 nM T84726 CM42CA 118728824 Ki > 4000 nM T84726 C9Q7CL 118728825 Ki > 4000 nM T84726 CCR3S0 118728826 Ki = 2700 nM T84726 CDC38O 134823958 IC50 = 450 nM T84726 CQ84IZ 136180335 Ki > 4000 nM T84726 C7ZE5Q 155511547 IC50 = 2230 nM T84726 CNF96Z 155519769 IC50 = 11.8 nM T84726 CI31SP 155527821 IC50 = 415 nM T84726 CET2B6 155531372 IC50 = 94 nM T84726 CS08FU 155533862 IC50 = 56 nM T84726 C8K3XJ 155537606 IC50 = 173 nM T84726 CDU52V 155538567 IC50 = 961 nM T84726 C2TMB4 155556732 IC50 = 963 nM T84726 CNH27R 155557555 IC50 = 7830 nM T84726 CL1MB0 155567304 IC50 = 802 nM T99295 D0J5VR 11625818 IC50 > 10000 nM T99295 D08QGT 17755052 IC50 > 10000 nM T99295 D0O6VZ 25254071 IC50 > 10000 nM T99295 C9U2YK 5109813 IC50 = 2511.89 nM T99295 C2IM0O 39733146 IC50 = 2511.89 nM T99295 C3VRO9 44557921 IC50 > 5888.44 nM T99295 CP2QD0 49784894 IC50 > 10000 nM T99295 CY36EH 51003592 IC50 = 630.96 nM T99295 CRJ5W8 51358113 IC50 > 10000 nM T99295 C7ZH0D 53308041 IC50 > 10000 nM T99295 C10YUH 53318615 IC50 = 2511.89 nM T99295 CO40ME 57404800 IC50 = 2.512 nM T99295 CQ5Z4S 57404801 IC50 = 1 nM T99295 C78YHO 57404804 IC50 = 3.981 nM T99295 CQ4E8N 57405149 IC50 = 1 nM T99295 CA8BT7 57405314 IC50 = 19.95 nM T99295 CI40MW 57405315 IC50 = 125.89 nM T99295 CGN72O 57405485 IC50 = 0.3162 nM T99295 C5B9XS 57406164 IC50 = 1.585 nM T99295 CEI2S9 57406702 IC50 = 5.012 nM T99295 C9Z1UL 57407079 IC50 = 0.7943 nM T99295 CHIU94 57545876 IC50 = 1.585 nM T99295 C3PL1S 66800530 IC50 = 100 nM T99295 CJN4M2 66806967 IC50 = 39.81 nM T99295 C5BZ2V 67981475 IC50 = 31.62 nM T99295 CK86XZ 67982080 IC50 = 10 nM T99295 CS0TY5 67982485 IC50 = 50.12 nM T99295 CE5OS6 67982535 IC50 = 15.85 nM T99295 C9A2RD 67982543 IC50 = 3981.07 nM T99295 C7A0GH 67982639 IC50 = 50.12 nM T99295 CW79LA 67982712 IC50 = 6.31 nM T99295 CUQ2W1 68095924 IC50 = 39.81 nM T99295 CUR8N0 68096082 IC50 = 10 nM T99295 CX65CB 71597290 IC50 = 450 nM T99295 CNX76A 72544842 IC50 = 1584.89 nM T99295 CBF70W 76310805 IC50 = 316.23 nM T99295 CM4N8A 76325342 IC50 = 630.96 nM T99295 C92ZAB 76325343 IC50 = 7943.28 nM T99295 CQ8YC1 76332568 IC50 = 5.012 nM T99295 CY3LO5 76336173 IC50 = 199.53 nM T99295 C9I7TY 78319187 IC50 = 6.31 nM T99295 CV6PI8 87562294 IC50 = 398.11 nM T99295 CK4Y2U 91758319 IC50 > 100000 nM T99295 C58XRY 122184465 IC50 = 158.49 nM T99295 C16ALM 122184466 IC50 = 100 nM T99295 CIX19J 122184467 IC50 = 1000 nM T99295 CDZY02 122184468 IC50 = 2511.89 nM T99295 CTH70U 122184469 IC50 = 79.43 nM T99295 C9ZXR7 122184470 IC50 = 630.96 nM T99295 CNJ9Z4 122184471 IC50 = 630.96 nM T99295 CMCP83 122184472 IC50 = 1584.89 nM T99295 CS41EG 122184473 IC50 = 1584.89 nM T99295 CZ36GL 122184474 IC50 = 15848.93 nM T99295 CU4ZT6 122184475 IC50 = 25118.86 nM T99295 C3H9PR 122184476 IC50 = 316.23 nM T99295 CU40TW 122184477 IC50 = 316.23 nM T99295 C8IK9C 122184478 IC50 = 3162.28 nM T99295 CAMD31 122184479 IC50 = 1258.93 nM T99295 C1F9RK 122184480 IC50 = 1000 nM T99295 C7XW1K 122184481 IC50 = 10000 nM T99295 CRUX54 122184482 IC50 = 15848.93 nM T99295 CQ7W0P 122184526 IC50 = 7943.28 nM T99295 CA5YB2 122184529 IC50 = 2511.89 nM T99295 C64YPH 122184530 IC50 = 12589.25 nM T99295 C4AGX5 122184531 IC50 = 3162.28 nM T99295 CQL4K5 122184532 IC50 = 1584.89 nM T99295 CRKV74 122184533 IC50 = 25118.86 nM T99295 CX14YD 122184534 IC50 = 7943.28 nM T99295 CM6A4S 122184535 IC50 = 630.96 nM T99295 CF86YS 122184536 IC50 = 158.49 nM T99295 CH08SN 122184537 IC50 = 501.19 nM T99295 CYRH97 122184538 IC50 = 316.23 nM T99295 CD4W0Z 122184539 IC50 = 630.96 nM T99295 CH8Y3Q 122184540 IC50 = 5.012 nM T99295 CDA85R 122184541 IC50 = 7.943 nM T99295 CF36XJ 122184542 IC50 = 39.81 nM T99295 CQ6O7H 122184543 IC50 = 1.995 nM T99295 CS4MN0 122184544 IC50 = 1 nM T99295 CEO76N 123131772 IC50 = 48000 nM T99295 CQP8L7 123131773 IC50 = 8190 nM T99295 C2OP5X 123131774 IC50 = 660 nM T99295 C8MSY6 134132647 IC50 = 12280 nM T99295 CZQ20R 134146889 IC50 = 17070 nM T99295 C2KU0W 134147646 IC50 = 553 nM T99295 C8ZPJ0 134150664 IC50 = 4860 nM T99295 CG8LE2 134151667 IC50 = 13400 nM T99295 C8NYC5 134155918 IC50 = 1128 nM T99295 C54FXD 134957362 IC50 > 10000 nM T99295 CV3UE9 137333450 IC50 = 574.1 nM T99295 C9O2PL 145958063 IC50 = 163.7 nM T99295 C9NS6T 145958690 IC50 = 130.6 nM T99295 D0H0HR 49836027 IC50 > 10000 nM T99295 D0P5TI 58441401 IC50 > 1000 nM T99295 D0S5YV 6852167 IC50 = 1100 nM T55709 D0G2XR 11239949 IC50 = 1920 nM T55709 C0US1F 764866 IC50 = 2600 nM T55709 CXM73B 2838414 IC50 = 1480 nM T55709 C8H1DV 2992288 IC50 > 300000 nM T55709 CY9DG1 10033990 IC50 = 1400 nM T55709 CMYK20 10078582 IC50 = 15000 nM T55709 C51WPX 10258491 IC50 = 37500 nM T55709 C0ORY6 10370410 IC50 = 300 nM T55709 C50GYQ 10484792 IC50 = 9600 nM T55709 C97PYO 10531232 IC50 > 1000000 nM T55709 CU48JT 10628095 IC50 = 80000 nM T55709 CVTP23 10652002 IC50 = 20000 nM T55709 CLW9R5 10722438 IC50 = 17000 nM T55709 C2G5DV 10723546 IC50 = 17000 nM T55709 CWJ3H8 10769646 IC50 = 100000 nM T55709 CT6OX2 10770264 IC50 = 1200 nM T55709 C2YK1V 10792844 IC50 = 100000 nM T55709 C62WNR 10792883 IC50 = 23000 nM T55709 C72QWY 10817558 IC50 = 136700 nM T55709 C5Y3MR 10864598 IC50 = 2100 nM T55709 C2JH9S 10973684 IC50 = 13200 nM T55709 C7NO9F 10984774 IC50 = 52800 nM T55709 CS16UM 11082270 IC50 = 84200 nM T55709 CD2SQ7 11158130 IC50 = 8800 nM T55709 CY5XP9 11158281 IC50 = 20600 nM T55709 C5EB1I 11158640 IC50 = 3000 nM T55709 C6UQ5O 11170373 IC50 = 1400 nM T55709 C42DMC 11192995 IC50 = 11100 nM T55709 CSJ1R4 11193161 IC50 = 1900 nM T55709 C0KL9U 11193856 IC50 = 4800 nM T55709 C1QX5Z 11205009 IC50 = 8400 nM T55709 CN75YR 11205032 IC50 = 1800 nM T55709 CH9CO5 11205090 IC50 = 1200 nM T55709 CI2O0L 11205213 IC50 = 96100 nM T55709 C5GM6Y 11216549 IC50 = 500 nM T55709 C2ZJY0 11216769 IC50 = 133000 nM T55709 C2GF6I 11227819 IC50 = 2900 nM T55709 CKO98J 11227850 IC50 = 400 nM T55709 C27DIS 11228087 IC50 = 1300 nM T55709 CL5S2X 11228090 IC50 = 9000 nM T55709 CF2N0X 11228315 IC50 = 2100 nM T55709 CSXF65 11238662 IC50 = 37700 nM T55709 C7T5IO 11251384 IC50 = 400 nM T55709 CNXU39 11251673 IC50 = 5700 nM T55709 CVK0U3 11262832 IC50 = 17800 nM T55709 CV0D3J 11262930 IC50 = 600 nM T55709 CE95KV 11297195 IC50 = 9600 nM T55709 CW7PF2 11297300 IC50 = 2200 nM T55709 CRC27V 11320058 IC50 = 10200 nM T55709 CFQ9N2 11320446 IC50 = 56800 nM T55709 C0T8DM 11331136 IC50 = 5800 nM T55709 C6HK4N 11331675 IC50 = 20600 nM T55709 CQY75R 11342615 IC50 = 81100 nM T55709 C7GCH3 11343599 IC50 = 11400 nM T55709 CIZ0B9 11355042 IC50 = 147000 nM T55709 CBD8A0 11366063 IC50 = 4300 nM T55709 CRSC54 11366263 IC50 = 1500 nM T55709 C8WA0K 11366336 IC50 = 19800 nM T55709 CISF61 11377969 IC50 = 11400 nM T55709 C7JNU4 11388209 IC50 = 11900 nM T55709 CEIU90 11399746 IC50 = 4400 nM T55709 CSQ4M9 11399908 IC50 > 200000 nM T55709 CJ1RW9 11400295 IC50 = 3100 nM T55709 C4XMJ3 11411692 IC50 = 9700 nM T55709 C0X5EL 11421622 IC50 = 24000 nM T55709 C4Q3KZ 11422543 IC50 = 39700 nM T55709 CTVD65 11422951 IC50 = 2300 nM T55709 C3QFZ9 11423157 IC50 = 46100 nM T55709 CC1B9D 11445422 IC50 = 63300 nM T55709 CB0J9Q 11457136 IC50 = 1000 nM T55709 CO2P4Z 11457348 IC50 = 57500 nM T55709 CVT3Y8 11480043 IC50 = 3500 nM T55709 CB7NS0 11480093 IC50 = 5700 nM T55709 CACS26 11561968 Ki > 10000 nM T55709 CU0E8O 11690457 Ki > 10000 nM T55709 C1MY3N 11763569 IC50 = 15000 nM T55709 CV2C5Y 11763720 IC50 > 200000 nM T55709 C56NAT 11766845 IC50 = 24800 nM T55709 CK7MR6 11787351 IC50 = 7200 nM T55709 C1X4EN 18525875 IC50 = 87000 nM T55709 CP0Q7H 18525904 IC50 > 2000000 nM T55709 C65VIL 22385756 IC50 > 300000 nM T55709 CNJ5Z6 44396626 IC50 > 100000 nM T55709 C9CGM8 44396644 IC50 = 48200 nM T55709 C41HZE 44396664 IC50 = 3400 nM T55709 CMOG56 44396710 IC50 > 100000 nM T55709 CKM7S8 44396762 IC50 > 100000 nM T55709 C7YM4V 44396776 IC50 = 98000 nM T55709 CMB29W 44396816 IC50 = 2600 nM T55709 C4N1QT 44423477 EC50 = 1300 nM T55709 CHO96M 52952144 IC50 = 780 nM T55709 C4JG6W 52952244 IC50 = 8430 nM T55709 CB7RH9 56839384 IC50 = 9650 nM T55709 CD12MJ 56839386 IC50 = 300 nM T55709 C0K2QT 56839388 IC50 = 1350 nM T55709 C48POV 56839584 IC50 = 2000 nM T55709 C4QT0F 56929921 IC50 = 4250 nM T55709 C5AWQ9 56929924 IC50 = 4400 nM T55709 C0IMN9 56930067 IC50 = 13500 nM T55709 C20PTZ 56930069 IC50 = 4200 nM T55709 CV4QP9 56930070 IC50 = 14200 nM T55709 CZW5Y9 56930212 IC50 = 12500 nM T55709 C3RK7Q 56930214 IC50 = 11600 nM T55709 CRQ97A 56930216 IC50 = 6150 nM T55709 CS8HX6 56930351 IC50 = 15000 nM T55709 CM6D5O 56932005 IC50 > 20000 nM T55709 CXWD86 56932007 IC50 = 17300 nM T55709 CHVY14 57392710 IC50 = 3100 nM T55709 C9VD3O 57396192 IC50 = 23800 nM T55709 C1MR8Q 60097495 IC50 > 10000 nM T55709 CUC7B3 66557964 IC50 > 50000 nM T55709 CSM71R 78425823 IC50 = 66 nM T55709 C5XIM6 86300181 IC50 = 1300 nM T55709 COZ3X2 86300470 IC50 = 4950 nM T55709 C1LD7C 86300475 IC50 = 1430 nM T55709 C1PC2W 86344482 IC50 = 17200 nM T55709 C1W7OE 90467110 IC50 = 1000 nM T55709 C19OKD 90467265 IC50 = 9560 nM T55709 CW3ST4 90666558 EC50 = 520 nM T55709 C5QX7D 102514724 IC50 = 920 nM T55709 C8U1RL 102596393 IC50 = 3900 nM T55709 C3DWX7 117609929 IC50 = 457 nM T55709 CYB35C 117609959 IC50 = 2600 nM T55709 C8GF6X 117610126 IC50 = 251 nM T55709 C15WYK 117610128 IC50 = 255 nM T55709 C75UFA 117610129 IC50 = 233 nM T55709 CSH1O2 117610137 IC50 = 85 nM T55709 C4Q3WV 117610193 IC50 = 268 nM T55709 CM3N0B 117610195 IC50 = 165 nM T55709 CNQ3E4 127025627 IC50 = 20 nM T55709 CS2KH3 129892324 IC50 = 1660 nM T55709 CZ6RE9 129892327 IC50 = 1630 nM T55709 CS1LN3 129892335 IC50 = 37540 nM T55709 C3NK6L 129892341 IC50 = 6850 nM T55709 CSWX10 129892346 IC50 = 2790 nM T55709 C5GZR2 129892349 IC50 = 2020 nM T55709 C46ZUJ 129892352 IC50 = 3270 nM T55709 CW9CG3 129892358 IC50 = 16220 nM T55709 CGVM05 129892359 IC50 = 9510 nM T55709 C54FXD 134957362 IC50 > 10000 nM T36959 D0E3TC 44259 IC50 = 850 nM T36959 D0MR0B 54766013 IC50 > 10000 nM T36959 CPQ31L 25195294 IC50 = 11.13 nM T36959 CN2QG1 44223357 IC50 = 26.5 nM T36959 CYH6P3 44520205 IC50 > 10000 nM T36959 CEA13T 46834838 IC50 = 770 nM T36959 CDV74N 50997747 IC50 = 27 nM T36959 C91FTP 57339386 IC50 = 52.4 nM T36959 CIP7B1 60182373 IC50 = 55 nM T36959 CQ6KV9 60182388 IC50 = 14.4 nM T36959 C91RWL 66561650 IC50 > 5000 nM T36959 CV63UL 67240318 IC50 > 10000 nM T36959 C2LD1B 121232401 IC50 = 4 nM T36959 CF4BN6 127050359 IC50 = 340 nM T36959 CGQH20 127050360 IC50 = 2300 nM T36959 CEB1O8 127050361 IC50 = 1000 nM T36959 C1NDK3 127050362 IC50 = 26 nM T36959 CDE6P8 127051209 IC50 = 120 nM T36959 CN2BE1 127051215 IC50 = 4600 nM T36959 C4R0JO 127051568 IC50 = 48 nM T36959 C2IL1U 127051569 IC50 = 800 nM T36959 CM9WR2 127051570 IC50 = 17 nM T36959 C41UTI 127051571 IC50 = 230 nM T36959 CR9OK4 127051572 IC50 = 940 nM T36959 CFU6S7 127053039 IC50 = 980 nM T36959 CI2YE9 132606873 IC50 = 62 nM T36959 CBP31D 137639641 IC50 = 1785 nM T36959 CK7AQ5 137645799 IC50 = 1256 nM T36959 CS61AX 137659496 IC50 > 100000 nM T36959 CPT0V7 138454752 IC50 = 51 nM T36959 C2MD1Q 155513187 IC50 > 10000 nM T36959 D05NEC 60182364 IC50 < 5 nM T36959 D06CMG 91754554 IC50 = 27 nM T36959 D0F2MP 60182389 IC50 < 5 nM T36959 D0PP6Y 60182393 IC50 = 42.1 nM T36959 D0RF7O 44577753 IC50 = 46 nM T36959 D0Y0BK 11524144 IC50 = 106.3 nM T44991 D0H2DQ 4912 IC50 > 50000 nM T44991 D0X1VJ 216325 IC50 = 6000 nM T44991 C4G2RM 7324 IC50 = 40000 nM T44991 C3XND9 9398 IC50 = 7000 nM T44991 CJY63Z 13655 IC50 = 11000 nM T44991 C45SBJ 16008 IC50 = 20000 nM T44991 C98CFG 20062 IC50 = 10000 nM T44991 C90NKY 41743 IC50 = 15000 nM T44991 C3L0BT 67300 IC50 = 10000 nM T44991 CM1O3C 67301 IC50 = 11000 nM T44991 CKL46X 85504 IC50 = 17000 nM T44991 CXFP15 85505 IC50 = 15000 nM T44991 CH6M4E 96924 IC50 = 5000 nM T44991 CKM1X8 128677 IC50 = 175 nM T44991 C3T4YX 296616 IC50 = 15000 nM T44991 C0DFY8 348301 IC50 = 5000 nM T44991 CXI3Y4 645569 IC50 > 100000 nM T44991 C5Q0FP 745480 IC50 = 59000 nM T44991 CYBV18 916176 IC50 = 18000 nM T44991 C16YNJ 962611 IC50 = 17000 nM T44991 CJ2IM5 2768393 IC50 = 4000 nM T44991 COB6U4 2807642 IC50 = 2500 nM T44991 C6S5DT 2833646 IC50 = 3000 nM T44991 CIG9B6 2842419 IC50 = 8000 nM T44991 CC9L3V 2899735 IC50 = 9000 nM T44991 CQ9F2K 3729614 IC50 = 8000 nM T44991 CXY7P4 5323285 IC50 = 10000 nM T44991 CH2S0W 7638374 IC50 = 5000 nM T44991 CEGN81 7749530 IC50 = 18000 nM T44991 CT3BF9 9797597 IC50 = 21000 nM T44991 C74QCT 9798233 IC50 > 4000 nM T44991 CCI90K 9799728 IC50 > 4000 nM T44991 C18UGE 9818339 IC50 = 20000 nM T44991 CJQ2W6 9835897 IC50 > 1000 nM T44991 C6G5RT 9836507 IC50 > 4000 nM T44991 CUGN49 9836683 IC50 > 1000 nM T44991 CJ5SU0 9839311 IC50 > 1000 nM T44991 CSK6P4 9841875 IC50 = 2700 nM T44991 C5DRX6 9856682 IC50 > 1000 nM T44991 C9MA3Z 9858009 IC50 = 23 nM T44991 C0ZQV7 9858022 IC50 = 770 nM T44991 C3MG0X 9860649 IC50 > 4000 nM T44991 C8IO4M 9878726 IC50 = 19000 nM T44991 C91VCO 9878930 IC50 = 11000 nM T44991 CP34JF 9879093 IC50 > 1000 nM T44991 C5S6CZ 9879529 IC50 = 3900 nM T44991 CBKH73 9880710 IC50 = 130 nM T44991 C1L5WE 9880711 IC50 > 1000 nM T44991 C0O5BM 9881984 IC50 = 39000 nM T44991 C0W1SB 9882382 IC50 = 65000 nM T44991 CY7KG3 9883504 IC50 = 70 nM T44991 CL1FR4 9900816 IC50 > 6 nM T44991 C3D1XN 9900943 IC50 > 1000 nM T44991 C9DHR2 9901085 IC50 = 850 nM T44991 CRND31 9901574 IC50 > 1000 nM T44991 CBM7Y3 9903965 IC50 = 2300 nM T44991 CKJ7T0 9903998 IC50 = 20000 nM T44991 C1JI7S 9904207 IC50 = 3500 nM T44991 C3VJ9K 9904395 IC50 > 4000 nM T44991 C62JUP 9904430 IC50 > 4000 nM T44991 CYN51E 9905179 IC50 > 4000 nM T44991 CDML85 9906347 IC50 = 20 nM T44991 CO63ID 9921367 IC50 = 2100 nM T44991 CQ4WG3 9921987 IC50 > 153 nM T44991 C9T3ME 9922373 IC50 > 4000 nM T44991 CO5L2R 9922793 IC50 > 100 nM T44991 C36KVQ 9922943 IC50 = 19000 nM T44991 CW5P9J 9924766 IC50 > 1000 nM T44991 C7QP1H 9944101 IC50 = 140 nM T44991 C2JZW5 9944163 IC50 > 1000 nM T44991 C9AJP0 9944774 IC50 > 200 nM T44991 CL9I6U 9945784 IC50 > 100 nM T44991 CB3P7T 9946091 IC50 > 1000 nM T44991 CYJ59B 9946991 IC50 = 79 nM T44991 CAFK13 9947244 IC50 > 4000 nM T44991 CR4LP3 9948282 IC50 = 15000 nM T44991 CNH47D 9948311 IC50 > 4000 nM T44991 C0YEQ7 9952465 IC50 > 1000 nM T44991 C2TYQ1 9953413 IC50 > 100000 nM T44991 CLMJ59 9960862 IC50 = 9000 nM T44991 C4QI0E 9961854 IC50 > 50000 nM T44991 CWH3L0 9965679 IC50 > 4000 nM T44991 CI4DU5 9966679 IC50 = 46000 nM T44991 CFEI36 9967126 IC50 > 4000 nM T44991 CA5W9Z 9967290 IC50 = 930 nM T44991 CS9DM3 9967511 IC50 > 1000 nM T44991 CYXW91 9968489 IC50 > 100 nM T44991 C1RUK3 10070771 IC50 = 4500 nM T44991 CX30HT 10089338 IC50 > 1000 nM T44991 CY23GM 10108997 IC50 > 1000 nM T44991 C2P4UO 10110987 IC50 > 4000 nM T44991 CTW3P9 10116693 IC50 = 170 nM T44991 C07COW 10132518 IC50 > 1000 nM T44991 C6N1FU 10134148 IC50 = 3500 nM T44991 CH49BD 10154440 IC50 > 1000 nM T44991 COF2S9 10154441 IC50 > 1000 nM T44991 CL7H2B 10154801 IC50 = 880 nM T44991 C0CP1T 10155661 IC50 = 470 nM T44991 CSB5F9 10156828 IC50 = 330 nM T44991 CF4DP2 10177047 IC50 = 370 nM T44991 C6RN4F 10178848 IC50 > 10 nM T44991 CHN3X1 10202790 IC50 > 4000 nM T44991 CD95KA 10221525 IC50 > 400 nM T44991 CJZU30 10267771 IC50 > 1000 nM T44991 C2OQ0K 10267925 IC50 > 1000 nM T44991 C9C0UG 10291112 IC50 > 4000 nM T44991 CWZU32 10291698 IC50 = 74 nM T44991 CTUP45 10291904 IC50 > 4000 nM T44991 CM05NG 10298900 IC50 = 420 nM T44991 C7KO6U 10361323 IC50 > 1000 nM T44991 CZ3DK8 10566084 IC50 = 10000 nM T44991 C5Q8EF 10566766 IC50 = 10000 nM T44991 CN3H5M 10632359 IC50 = 1300 nM T44991 C6QZG3 10686899 IC50 > 4000 nM T44991 CZF1H3 10708446 IC50 > 4000 nM T44991 CAPG02 10732433 IC50 > 1000 nM T44991 C6K5GC 10860379 IC50 > 1000 nM T44991 CSO95L 10862219 IC50 > 1000 nM T44991 C7OFZ9 10863087 IC50 > 1000 nM T44991 C6PRJ8 10880644 IC50 = 64 nM T44991 CV9I3D 10891751 IC50 = 85 nM T44991 C9X6VP 10892285 IC50 = 780 nM T44991 C9DUB8 10892642 IC50 > 1000 nM T44991 CS1T3C 10896625 IC50 > 1000 nM T44991 CARC06 10904579 IC50 > 180 nM T44991 CHWL69 10905666 IC50 > 140 nM T44991 CLPA31 10906508 IC50 > 1000 nM T44991 C7YG6L 10924566 IC50 = 191 nM T44991 CR51AV 10970154 IC50 = 5 nM T44991 CQ6E7Y 10970207 IC50 > 1000 nM T44991 CB31OE 10980658 IC50 > 1000 nM T44991 C94UAC 10982608 IC50 = 20 nM T44991 CVR4Y3 11001541 IC50 > 1000 nM T44991 CCP7K5 11013542 IC50 > 1000 nM T44991 C1ZRL6 11014018 IC50 = 6 nM T44991 CIW6J5 11023935 IC50 > 24 nM T44991 C7NCE4 11036406 IC50 > 1000 nM T44991 CM5HI8 11045962 IC50 = 17 nM T44991 C7U2JK 11048059 IC50 > 1000 nM T44991 C7E6GN 11048585 IC50 > 1000 nM T44991 CNHY70 11057712 IC50 > 1000 nM T44991 COE6W0 11068095 IC50 = 19 nM T44991 C9Q0MP 11070710 IC50 > 1000 nM T44991 CZSV01 11078679 IC50 > 1000 nM T44991 C1KE2T 11079237 IC50 > 1000 nM T44991 C8SRX4 11080157 IC50 > 1000 nM T44991 C5T1BO 11089640 IC50 > 1000 nM T44991 CQYV18 11091464 IC50 > 1000 nM T44991 CSF94U 11102008 IC50 > 1000 nM T44991 C51PTF 11109642 IC50 = 91 nM T44991 C8RF0J 11111846 IC50 > 1000 nM T44991 C8WI4X 11120977 IC50 > 1000 nM T44991 CUGV75 11122788 IC50 > 1000 nM T44991 CHIT70 11134430 IC50 > 1000 nM T44991 CRPC48 11134652 IC50 > 1000 nM T44991 C5DUF4 11760748 IC50 > 1000 nM T44991 C8BJ0L 11783098 IC50 = 240 nM T44991 C43LZD 11783922 IC50 > 1000 nM T44991 CKRM28 11793014 IC50 > 4000 nM T44991 CLX8Z9 11825588 IC50 > 1000 nM T44991 C7SG8X 11828434 IC50 > 1000 nM T44991 CE0I5U 14622573 IC50 = 19000 nM T44991 C2A0PI 18670114 IC50 = 2500 nM T44991 C1NYZ2 43213376 IC50 = 10000 nM T44991 C5CUX9 43265835 IC50 = 15000 nM T44991 C36WMA 44264201 IC50 > 4000 nM T44991 C0TE8R 44296991 IC50 = 5000 nM T44991 CH28OX 44297034 IC50 = 6000 nM T44991 C8KS4V 44297035 IC50 = 7000 nM T44991 C9WRD5 44297075 IC50 = 30000 nM T44991 C51MSD 44297089 IC50 = 10000 nM T44991 CU8OV5 44297227 IC50 = 7000 nM T44991 CNXU32 44319091 IC50 = 20000 nM T44991 CEY12S 44319174 IC50 = 25000 nM T44991 C2WQ4O 44319200 IC50 = 100000 nM T44991 CDE74L 44319212 IC50 = 30000 nM T44991 CVA0S4 44319255 IC50 > 50000 nM T44991 CR0S8D 44319289 IC50 = 40000 nM T44991 C2CXV6 44319428 IC50 = 45000 nM T44991 CVP86T 44319432 IC50 = 30000 nM T44991 C8TBZ2 44319572 IC50 = 17000 nM T44991 CO1W7G 44319600 IC50 = 8000 nM T44991 C8X5EI 44319601 IC50 = 110000 nM T44991 CTJ7M3 44319636 IC50 = 37000 nM T44991 CH2W8G 44319651 IC50 = 40000 nM T44991 CEF0J7 44319652 IC50 = 55000 nM T44991 CM7P9U 44344139 IC50 > 1000 nM T99524 D03RZV 5504 Ki = 1640 nM T99524 D0H0HJ 19493 EC50 = 1510 nM T99524 D0L4HY 5702063 EC50 = 90 nM T99524 D0P6UB 10836 EC50 = 1300 nM T99524 D0P8RS 6178111 EC50 > 10000 nM T99524 D0T3LF 5826 EC50 = 140 nM T99524 D0U0RZ 4771 EC50 = 5470 nM T99524 D0KC5X 10468498 EC50 = 15 nM T99524 CH8TW2 4653 EC50 = 740 nM T99524 C4Y7PS 4657 EC50 = 5980 nM T99524 CRD7M3 11492 EC50 = 1740 nM T99524 C08ENH 11503 EC50 = 250 nM T99524 C6IM0L 15006 EC50 > 10000 nM T99524 C43RNM 15651 EC50 = 1792 nM T99524 C9F3EI 19933 EC50 > 10000 nM T99524 CA75NH 25125 EC50 = 1490 nM T99524 C2MO8K 29669 EC50 = 1000 nM T99524 CP07AC 36604 EC50 = 3300 nM T99524 C0F5BM 67430 EC50 = 2860 nM T99524 C39DLT 70287 EC50 = 5050 nM T99524 CUEX90 73874 EC50 = 5030 nM T99524 C4J1XQ 74865 EC50 = 614 nM T99524 C1BJ8Y 74866 EC50 = 1444 nM T99524 C4VQ6L 74896 EC50 = 144 nM T99524 C5Q8JB 76632 EC50 = 2010 nM T99524 C6NUX9 76751 EC50 = 4380 nM T99524 CI86XG 83117 EC50 = 77 nM T99524 CQB5G7 95153 EC50 = 167386 nM T99524 CQ85KD 104223 EC50 = 3950 nM T99524 CE04WR 120234 EC50 = 1040 nM T99524 CGVM59 123528 Ki = 500 nM T99524 CXG98M 135740 EC50 = 6478 nM T99524 CLP01Z 139381 EC50 = 189 nM T99524 CJ7V6U 144047 EC50 = 9100 nM T99524 CQK3J6 151465 EC50 = 3460 nM T99524 CH37LO 176468 EC50 = 687 nM T99524 C8YMA9 176469 EC50 = 5980 nM T99524 C6Y4MO 210602 EC50 = 7880 nM T99524 C0ESJ5 210890 EC50 = 1380 nM T99524 CE78TU 211415 EC50 = 377 nM T99524 CCQ34V 217958 EC50 = 3430 nM T99524 CV7YM6 240539 Ki = 400 nM T99524 C1OHP9 410085 EC50 = 638 nM T99524 CY1L8V 533915 EC50 = 1540 nM T99524 C3ATE2 533928 EC50 = 150 nM T99524 CC72JQ 594090 Ki = 20 nM T99524 C5V9NS 643357 EC50 = 65 nM T99524 CM4N8J 644000 EC50 = 2960 nM T99524 C97QDH 800907 EC50 > 100000 nM T99524 C80GSE 854031 EC50 = 370 nM T99524 C41RLK 1547949 EC50 = 361 nM T99524 C5U9ZB 1547950 EC50 = 129 nM T99524 C4EZW6 1988106 EC50 = 11600 nM T99524 CKT5V4 2063868 EC50 = 355 nM T99524 CC6Y2H 2730263 EC50 > 10000 nM T99524 C36PNS 2734091 EC50 = 57 nM T99524 CRYX58 2734094 EC50 = 312 nM T99524 CQ1D7C 2734101 EC50 = 51 nM T99524 CNK78J 2734758 EC50 = 1160 nM T99524 C56ZPJ 2735689 EC50 = 5112000 nM T99524 C39XKS 2942630 IC50 = 3790 nM T99524 CH8P2E 3046161 EC50 = 11730 nM T99524 C1ER5D 3050061 EC50 = 6570 nM T99524 CK5GP3 3151733 EC50 = 18100 nM T99524 CDFX53 3151734 EC50 > 100000 nM T99524 CU6VY0 3413972 EC50 > 100000 nM T99524 CXE8N9 5338725 EC50 > 100000 nM T99524 CSV0T2 5356927 EC50 > 100000 nM T99524 CZ3DA6 7021736 EC50 = 398 nM T99524 CL4XC0 9561656 EC50 > 100000 nM T99524 C1ASI4 9563628 EC50 = 1230 nM T99524 C9QW6K 9568045 EC50 = 170 nM T99524 CC2X6K 9880217 EC50 = 9950 nM T99524 CU5KS9 10514616 EC50 = 103 nM T99524 CF19LK 10583272 EC50 = 501 nM T99524 CK0DL4 10678801 Ki = 4250 nM T99524 C84GAL 10751802 EC50 = 24400 nM T99524 CDU3B2 11116360 EC50 = 67 nM T99524 CIXA52 11252272 Ki = 2 nM T99524 CF2S1E 11426470 EC50 = 1200 nM T99524 CT38DB 11964124 EC50 = 205 nM T99524 CQI94M 11971703 EC50 = 3000 nM T99524 CWT52K 12234986 EC50 = 3160 nM T99524 CT9LI0 12351385 EC50 = 160 nM T99524 C3KC0R 12467520 EC50 = 630000 nM T99524 CL3S9X 12626561 EC50 = 31940 nM T99524 CKR86V 13178307 Ki = 65 nM T99524 C93YAC 13589773 EC50 = 7430 nM T99524 CZFP26 15581127 Ki = 36 nM T99524 C4GS3B 17809391 EC50 = 19100 nM T99524 CN4CL2 18349589 Ki = 138 nM T99524 C3ONZ7 18367548 EC50 = 8300 nM T99524 CR8V5U 18367556 EC50 = 6540 nM T99524 CDJY05 18954858 Ki = 1390 nM T99524 C16PQS 21742268 EC50 = 1800 nM T99524 CNVY52 21886837 EC50 = 530 nM T99524 C4UAK0 21887195 EC50 = 117 nM T99524 C17FZA 22072874 EC50 = 4320 nM T99524 C0U2SC 22072908 EC50 = 1290 nM T99524 CRNM25 22809970 EC50 = 6500 nM T99524 C1A9EF 23983765 EC50 = 15340 nM T99524 C9HR3G 24066917 EC50 = 5020 nM T99524 C9U8RQ 24729233 EC50 = 6410 nM T99524 C6K0IY 24771985 Ki = 4 nM T99524 CRU7Q0 24781714 Ki = 300 nM T99524 CEQY61 24781869 Ki = 24 nM T99524 COP87F 24894367 Ki = 68 nM T99524 C2ISG3 24946957 Ki = 48 nM T99524 C83AGK 24946958 Ki = 11 nM T99524 CE7LJ0 24946961 EC50 = 6.8 nM T99524 C0Q4AR 24946962 Ki = 11 nM T99524 CRS3C2 24946964 Ki = 4 nM T99524 CB5U0Y 24947139 Ki = 5 nM T99524 CX0T4Y 24947142 Ki = 6 nM T99524 C69PWD 24947144 Ki = 4 nM T99524 C3HA0Z 24947327 Ki = 13 nM T99524 C7JI0V 24948458 Ki = 2 nM T99524 C6E1PS 24952246 Ki = 12 nM T99524 CY9C3Z 24956883 Ki = 35 nM T99524 CNI67V 24963281 EC50 = 18 nM T99524 C2UT1W 24963283 EC50 = 330 nM T99524 CB68JF 24963286 EC50 = 18 nM T99524 C4PX5Z 24963287 EC50 = 2260 nM T99524 COZ8D3 24966106 EC50 = 23 nM T99524 CL71DQ 24966108 EC50 = 143 nM T99524 CM90WQ 24966113 EC50 = 31 nM T99524 CWJ72D 24966115 EC50 = 150 nM T99524 CPZ04W 24966469 EC50 = 165 nM T99524 C67BUG 24966828 EC50 = 2670 nM T99524 CZM6R8 25016282 EC50 = 580 nM T99524 C5ELY7 25016537 EC50 = 230 nM T99524 CFI04Q 25016800 EC50 = 29 nM T99524 C5U3HS 28635005 EC50 = 51600 nM T99524 CPCV49 29979100 EC50 = 3750 nM T99524 C6RQ7E 40578307 EC50 = 1900 nM T99524 C5YB3Q 43142643 EC50 > 100000 nM T99524 CH74WR 43142687 EC50 = 12100 nM T99524 CY5I7L 44370261 Ki = 32 nM T99524 CJRP90 44578414 EC50 = 1400 nM T99524 CX3B2T 44578415 EC50 = 767 nM T99524 C16RDN 44578545 EC50 = 1070 nM T99524 CLV98W 53318231 IC50 > 10000 nM T99524 C30SQT 54333224 EC50 = 330 nM T99524 C70GHX 56835991 EC50 = 17 nM T99524 C61WPO 57667099 EC50 = 140 nM T99524 C8S4KM 57667121 EC50 = 27 nM T99524 CE2J5X 58951676 Ki = 43000 nM T99524 CPNY90 58951824 Ki = 630 nM T99524 C1WB3P 58951908 Ki = 825 nM T99524 CTXV70 59173125 EC50 = 9 nM T99524 CVZ62F 59323617 EC50 = 490 nM T99524 CCT1S8 59323636 EC50 = 360 nM T99524 CA3K6C 59323671 EC50 = 154 nM T99524 C1P9EY 59323703 EC50 = 270 nM T99524 C7QV8M 59323754 EC50 = 21 nM T99524 CIA1R6 59323758 EC50 = 67 nM T99524 CY5SI4 59323783 EC50 = 12 nM T99524 CGV2H4 59323794 EC50 = 26 nM T99524 C37HLG 59323798 EC50 = 27 nM T99524 C8FDS2 59323824 EC50 = 2900 nM T99524 C1ZAX8 59323826 EC50 = 41 nM T99524 CXI2U9 59323836 EC50 = 1950 nM T99524 CJM74O 59323844 EC50 = 730 nM T99524 C4GAD8 59323854 EC50 = 1540 nM T99524 CG7T4Y 59323872 EC50 > 10000 nM T99524 C3WH6B 59708951 Ki = 470 nM T99524 CQ0F5Y 59708955 Ki = 1270 nM T99524 C82DUV 59728040 Ki = 40 nM T99524 C0YR8D 59728062 Ki = 80 nM T99524 CRC85H 59728070 Ki = 84 nM T99524 CPWN07 59728103 Ki = 12 nM T99524 CA8ZN6 59728125 Ki = 69 nM T99524 CH46FS 59728128 Ki = 12 nM T99524 CZJP48 59728187 Ki = 100 nM T99524 CJR0X2 59728194 Ki = 195 nM T99524 CVYR16 59728203 Ki = 100 nM T99524 C7BIF0 59728210 Ki = 128 nM T99524 CJTP70 59728229 Ki = 18 nM T99524 C1L0SB 59728233 Ki = 33 nM T99524 C8J3FP 59824833 EC50 = 27 nM T99524 C8FD3Y 66552052 Ki = 710 nM T99524 CS2LE8 66552123 Ki = 13300 nM T99524 CC6KW3 83032501 EC50 = 1600 nM T99524 C6IZX3 83034883 EC50 = 7000 nM T99524 C8ALY7 127031959 EC50 = 11 nM T99524 CRMH51 137633284 EC50 = 4900 nM T99524 CXZ7A6 145950350 EC50 = 11400 nM T99524 D02EPZ 24782016 Ki = 82 nM T99524 D05GOP 25175634 Ki > 5000 nM T99524 D07BAH 32893 EC50 = 250 nM T99524 D0C5RZ 5610 EC50 = 731 nM T99524 D0C7FL 77575 EC50 = 3400 nM T99524 D0HR1V 9950514 EC50 = 1510 nM T99524 D0O9ZY 25016538 EC50 = 59 nM T99524 D0Q6PI 1001 EC50 = 106 nM T99524 D0U3GZ 98527 EC50 = 7190 nM T57700 D00STL 644241 IC50 < 10 nM T57700 D01PZD 5329098 IC50 = 35 nM T57700 D04LVK 57379345 IC50 = 2855 nM T57700 D07NVU 9829523 IC50 = 109 nM T57700 D08CDI 208908 IC50 > 200000 nM T57700 D09GDD 11167602 IC50 = 6.1 nM T57700 D0AZ3C 5291 IC50 = 16.4 nM T57700 D0E6XR 3062316 IC50 = 2.6 nM T57700 D0G6QF 3081361 IC50 = 343 nM T57700 D0H0EQ 24826799 IC50 = 1.7 nM T57700 D0IQ6P 25102847 IC50 = 4 nM T57700 D0J9ZR 4477 IC50 = 27800 nM T57700 D0OB0F 5328940 IC50 = 181 nM T57700 D0R0MW 5329102 IC50 = 0.7 nM T57700 D0U3SY 49806720 IC50 > 5000 nM T57700 D0W5HK 216239 IC50 = 10 nM T57700 D02RJY 11442891 IC50 = 407 nM T57700 D02UFQ 11620908 IC50 > 10000 nM T57700 D03AND 11656518 IC50 = 20 nM T57700 D03HUX 49792852 IC50 > 10000 nM T57700 D03LWG 53235510 IC50 = 750 nM T57700 D06DMQ 59472121 Ki = 39 nM T57700 D07EHV 44814409 IC50 > 10000 nM T57700 D07HPJ 11476171 IC50 = 6300 nM T57700 D07HRU 9549295 IC50 = 4330 nM T57700 D09TAB 25151352 IC50 = 27 nM T57700 D0D1GF 42642645 IC50 = 4 nM T57700 D0E3TC 44259 IC50 = 3.6 nM T57700 D0M0XB 10302451 IC50 = 200 nM T57700 D0M9QZ 11485656 IC50 = 14 nM T57700 D0N8RV 9868037 IC50 = 10 nM T57700 D0O0LS 25141092 IC50 > 1000 nM T57700 D0O6WV 24794418 IC50 = 144 nM T57700 D0P1CV 46191454 IC50 > 10000 nM T57700 D0P6DJ 151194 IC50 = 730 nM T57700 D0Q9UX 16718576 IC50 = 668 nM T57700 D0S7HM 16041424 IC50 = 120 nM T57700 D0Z6MT 16662431 IC50 = 2 nM T57700 D03BNU 59604787 IC50 > 3500 nM T57700 D0H4GI 10275001 IC50 = 57 nM T57700 D0IT6Q 3038522 IC50 = 170 nM T57700 D0T3ME 156422 IC50 > 30000 nM T57700 CB1VW3 1400 IC50 = 1318 nM T57700 CWH85P 42723 IC50 = 400 nM T57700 CZF80A 72035 IC50 = 10 nM T57700 CK50LA 149478 IC50 = 600 nM T57700 C2TGS4 149480 IC50 < 10 nM T57700 C6Y9CV 151193 IC50 = 620 nM T57700 CK0L4O 442514 IC50 = 2700 nM T57700 C1ZG2U 449087 IC50 > 10000 nM T57700 CFG1A0 732043 IC50 = 1400 nM T57700 CHC5I0 2971839 IC50 > 10000 nM T57700 CFY1D0 2974957 IC50 > 10000 nM T57700 C2DG6J 3068873 IC50 = 2500 nM T57700 CN4V2F 5320438 IC50 = 600 nM T57700 C52MYD 5327893 IC50 > 1000 nM T57700 CQ0ZP3 5327897 IC50 > 1000 nM T57700 C7KIT4 5327898 IC50 > 1000 nM T57700 CDK3J0 5703619 IC50 = 10 nM T57700 C6L5HS 6419386 IC50 > 10000 nM T57700 C3CQW0 6419387 IC50 = 2500 nM T57700 CWOA63 6419388 IC50 = 1000 nM T57700 CZVU64 6419389 IC50 = 1400 nM T57700 C9FN4B 6419390 IC50 = 3000 nM T57700 CN53YW 6419391 IC50 = 7900 nM T57700 C17NWJ 6419392 IC50 = 700 nM T57700 C13IRC 6419393 IC50 = 3500 nM T57700 C4FLE9 6419394 IC50 = 2000 nM T57700 C4GHT0 6419395 IC50 = 2700 nM T57700 C8SAQ1 6419396 IC50 > 10000 nM T57700 CP71CL 6419397 IC50 > 10000 nM T57700 CTZ4W0 6539971 IC50 = 32 nM T57700 CAOU70 6539972 IC50 = 8.913 nM T57700 CE9L8Y 6539983 IC50 = 28 nM T57700 CUPQ08 6539985 IC50 = 6 nM T57700 CK9TD3 6539988 IC50 = 67.61 nM T57700 CDA25S 6539989 IC50 = 83.18 nM T57700 C6Q4ZY 6539990 IC50 = 50 nM T57700 C3SXL8 6539991 IC50 = 19 nM T57700 CWC68D 6539992 IC50 = 15 nM T57700 CK23SV 6539994 IC50 = 26.92 nM T57700 C9ZN6H 6539995 IC50 = 33 nM T57700 C39QGE 6539996 IC50 = 109.65 nM T57700 C8EJI1 6539997 IC50 = 21.88 nM T57700 CYQ9D4 6539998 IC50 = 28.84 nM T57700 CH2EV5 6539999 IC50 = 50 nM T57700 C9GMT4 6540000 IC50 = 47.86 nM T57700 CWA5M6 6540001 IC50 = 141.25 nM T57700 C3SAD6 6540002 IC50 = 42.66 nM T57700 CU14NK 6540003 IC50 = 19 nM T57700 CIC64F 6540004 IC50 = 175 nM T57700 CMEZ23 6540005 IC50 = 181.97 nM T57700 CG1L6R 6540006 IC50 = 160 nM T57700 C92OFS 6540007 IC50 = 398.11 nM T57700 C7H4QP 6540008 IC50 = 930 nM T57700 CF97JX 6540009 IC50 = 580 nM T57700 C52OIP 6540010 IC50 = 800 nM T57700 C2O4MX 6540012 IC50 = 81.28 nM T57700 CSGQ06 6540015 IC50 = 790 nM T57700 CP32OT 6540016 IC50 = 954.99 nM T57700 C4NWO7 6540017 IC50 = 37.15 nM T57700 C8AU3M 6540018 IC50 = 360 nM T57700 C3K7TM 6540019 IC50 = 25.7 nM T57700 CM1TH0 6540020 IC50 = 810 nM T57700 CK19HQ 6540021 IC50 = 27 nM T57700 CXK07R 6540022 IC50 = 199.53 nM T57700 CFLH24 6540023 IC50 = 180 nM T57700 CJ17TA 6540024 IC50 = 38 nM T57700 C0BQ2E 6540025 IC50 = 54 nM T57700 CIUP42 6540026 IC50 = 28 nM T57700 CG17TN 6914611 IC50 = 26200 nM T57700 C7E2QK 6914613 IC50 > 50000 nM T57700 C6U8FR 8016699 IC50 = 500 nM T57700 CB9ZH4 9805421 IC50 = 421 nM T57700 C1E2DV 9826083 IC50 > 10000 nM T57700 CX10KR 9828962 IC50 = 110 nM T57700 CC90FJ 9869737 IC50 = 293 nM T57700 CHF7G5 9890746 IC50 = 220 nM T57700 C3EUB4 9911005 IC50 = 390 nM T57700 C1BZ0P 9928737 IC50 = 12 nM T57700 C26QHZ 10005638 IC50 > 10000 nM T57700 CYX27A 10006987 IC50 = 235 nM T57700 CMZ2S8 10029735 IC50 = 766 nM T57700 CUJR40 10062694 EC50 = 4 nM T57700 CEKL46 10070245 IC50 = 491 nM T57700 C2P6HN 10071040 IC50 > 1000 nM T57700 C8G5RH 10095463 IC50 > 1000 nM T57700 CIV15Q 10113978 IC50 = 74 nM T57700 C5WCL2 10117540 IC50 = 190 nM T57700 CP95FO 10181075 IC50 = 245 nM T57700 C3ER4N 10187285 IC50 = 6 nM T57700 CD7J3O 10231458 IC50 = 60 nM T57700 CAE03L 10231813 IC50 = 21 nM T57700 C7SFI1 10296883 IC50 > 10000 nM T57700 CC4G8B 10302519 IC50 = 4 nM T57700 C4FP8M 10303591 IC50 = 16 nM T57700 CUN52O 10345191 IC50 = 239 nM T57700 CDS29Z 10366675 IC50 > 1000 nM T57700 C6ZF0X 10386217 IC50 = 800 nM T57700 CA8B5T 10390073 IC50 > 10000 nM T57700 CU4R9M 10413666 IC50 > 1000 nM T57700 C7HBP6 10429593 IC50 > 10000 nM T57700 CSAZ29 10454329 IC50 > 1000 nM T57700 C95LYF 10457505 IC50 = 130 nM T57700 CY9DS7 10458235 IC50 > 1000 nM T57700 CJ4P5T 10905857 IC50 = 480 nM T57700 CJ05CL 11048367 IC50 = 50 nM T57700 C03XHM 11152545 IC50 = 5 nM T57700 CW6Z5P 11154134 IC50 = 41 nM T57700 CB47NS 11156401 IC50 = 71 nM T57700 CU53KH 11177394 IC50 = 23440 nM T57700 C7ZB5L 11177668 IC50 = 69 nM T57700 CNG8F1 11178869 IC50 = 290 nM T57700 C6H5VA 11189551 IC50 = 102 nM T57700 CSWR60 11223082 IC50 = 790 nM T57700 CT0C5R 11235290 IC50 = 114 nM T57700 C8CF1H 11244819 IC50 = 44 nM T57700 C1Y7DB 11245809 IC50 = 5 nM T57700 CD9T6R 11257328 IC50 = 4 nM T57700 CJFX60 11259128 IC50 = 39 nM T57700 CV18PX 11265647 IC50 = 4443 nM T57700 CJ23CR 11268446 IC50 = 11 nM T57700 CBQ10L 11268741 IC50 = 42 nM T57700 CQL3P9 11271710 IC50 = 50 nM T57700 CI1H5P 11280431 IC50 = 14 nM T57700 CC24PZ 11281789 IC50 = 2630 nM T57700 CBOP58 11293798 Ki > 10000 nM T57700 C60ISR 11304968 IC50 = 339 nM T57700 CYK15J 11314310 IC50 = 17 nM T57700 CLX54H 11317348 IC50 = 40 nM T57700 CL7G8F 11325920 IC50 = 7 nM T57700 CI75ZE 11327388 IC50 = 27 nM T57700 CY54IT 11337407 IC50 = 21 nM T57700 CK1P7Y 11337894 IC50 = 13 nM T57700 CUT16W 11340683 IC50 = 53 nM T57700 C26BZX 11362471 Ki > 10000 nM T57700 CY8AQ4 11371508 IC50 = 42 nM T57700 CMN14Z 11373591 IC50 = 7 nM T57700 C25ZCN 11374110 IC50 = 56 nM T57700 CM30TC 11387552 IC50 < 10 nM T57700 CWXB93 11397177 Ki > 10000 nM T57700 CNT8W2 11404903 IC50 = 850 nM T57700 CPIM91 11406239 IC50 = 23 nM T57700 C6EP7S 11407183 IC50 = 24 nM T57700 CL7I5H 11407736 IC50 = 150 nM T57700 C6ML4B 11417108 IC50 = 34 nM T57700 C5KR0Y 11417521 IC50 = 12 nM T57700 CI34BN 11428396 IC50 = 15 nM T57700 CL9J6B 11428773 IC50 = 5 nM T57700 C6LJR3 11429321 IC50 = 216 nM T57700 CREQ51 11429654 IC50 = 43 nM T57700 CY0A4E 11429729 IC50 = 72 nM T57700 C5KG7W 11440661 IC50 = 14 nM T57700 CAM63T 11451774 IC50 = 10 nM T57700 CD97KV 11462058 IC50 = 18 nM T57700 CJ94MR 11465254 IC50 = 400 nM T57700 CN20YG 11465676 IC50 = 114 nM T57700 CJ2BH4 11473904 IC50 = 20 nM T57700 CK3M0T 11495270 IC50 = 7 nM T57700 CRJ3H2 11495362 IC50 = 19 nM T57700 CMIT06 11496035 IC50 = 303 nM T57700 CRU9D3 11508262 Ki = 46 nM T57700 C2T8YD 11511361 IC50 = 12 nM T57700 C8AY3B 11518031 IC50 < 25 nM T57700 C9DV1X 11525218 IC50 < 30 nM T57700 C98ENG 11525727 IC50 = 202 nM T57700 CL7X4Q 11530963 IC50 = 1900 nM T57700 COJI59 11539040 IC50 = 22 nM T57700 CTG83F 11539329 Ki > 1200 nM T57700 CD4LG5 11545419 IC50 = 16 nM T57700 C0OHL1 11561411 IC50 = 25 nM T57700 CACS26 11561968 Ki > 2000 nM T57700 CPW27V 11581044 Ki = 27 nM T57700 C9CDX4 11583287 IC50 = 153 nM T57700 CEM6P4 11583341 IC50 = 5 nM T57700 CI5W0C 11583439 IC50 = 938 nM T57700 C3VUO7 11588815 IC50 = 7 nM T57700 CA2KX0 11590078 IC50 = 12 nM T57700 CMIL86 11590363 Ki > 1200 nM T57700 C28FJS 11597486 IC50 = 3 nM T57700 C69FYK 11604142 Ki < 1 nM T57700 CQ5NP2 11604829 IC50 < 30 nM T57700 C8YIS9 11604883 IC50 = 25 nM T57700 CZD5J8 11605467 IC50 = 38 nM T57700 CJU5W6 11611103 Ki = 148 nM T57700 C8IKG5 11616255 IC50 = 500 nM T57700 C5B3XJ 11620410 IC50 = 30 nM T57700 CK34LS 11632737 IC50 = 370 nM T57700 CS2K5N 11634109 IC50 = 16 nM T57700 CYL45U 11634544 IC50 = 23 nM T57700 CFM2Y4 11640405 IC50 = 27 nM T57700 C9T6SC 11640926 Ki > 1200 nM T57700 CQ4OC2 11654378 IC50 = 3.5 nM T57700 C08DMH 11655667 IC50 = 233 nM T57700 CO52CP 11656170 IC50 = 637 nM T57700 CQ47BI 11662314 IC50 = 43 nM T57700 CU0E8O 11690457 Ki > 2000 nM T57700 C2CM0L 11690679 IC50 = 69 nM T57700 CSIN39 11690947 IC50 = 80 nM T57700 C4WM6K 11697289 IC50 = 3 nM T57700 CQ2P3D 11704845 IC50 = 5 nM T57700 CAL4G1 11705461 IC50 = 7 nM T57700 C9P0VD 11729539 IC50 = 360 nM T57700 CU5V9K 11749082 IC50 = 37 nM T57700 C9JT4S 11847343 IC50 = 35 nM T57700 CAZS08 11848309 IC50 = 421 nM T57700 C43IVN 11848567 IC50 = 149 nM T57700 C9LAY8 11848825 IC50 = 2007 nM T57700 CN1U7P 11855937 IC50 = 62 nM T57700 CYA0X2 11856199 IC50 = 36 nM T57700 C0A9WL 11856200 IC50 = 166 nM T57700 CJ5G9Y 11856201 IC50 = 50 nM T57700 COLP81 11856204 IC50 = 23 nM T57700 CSRQ05 11856467 IC50 = 64 nM T57700 CA2BL5 11856735 IC50 = 294 nM T57700 CI39TK 12004372 IC50 = 10500 nM T57700 CST0F3 12733993 IC50 = 250 nM T57700 C24FXN 15941243 IC50 = 3022 nM T57700 CG5IO2 15941244 IC50 = 91 nM T57700 C8Y1XP 15941246 IC50 = 6 nM T57700 CB94LR 15941247 IC50 = 37 nM T57700 CZ38JG 15941390 IC50 = 12 nM T57700 CE57UJ 15941392 IC50 = 11 nM T57700 C1AIM6 15941393 IC50 = 50 nM T57700 CN7PO9 15941394 IC50 = 18 nM T57700 C9E3RP 15941395 IC50 = 22 nM T57700 CSBF70 15941529 IC50 = 35 nM T57700 CQM93O 15941530 IC50 = 28 nM T57700 C7LB4I 15949613 IC50 = 170 nM T57700 CFPW41 16007116 Ki > 1200 nM T57700 CQI0A5 16043229 IC50 = 18 nM T57700 CZKD04 16043241 IC50 = 11 nM T57700 C9X4TQ 16043242 IC50 = 7 nM T57700 CZK8V6 16043304 IC50 = 110 nM T57700 C9JK2M 16059071 IC50 = 28 nM T57700 CW6UJ9 16059338 IC50 = 56 nM T57700 CH7MS6 16059729 IC50 = 20 nM T57700 CFKE48 16064750 IC50 = 20 nM T57700 CU5Y7N 16101466 IC50 = 11 nM T57700 C1U8XW 16109036 IC50 = 2800 nM T57700 C1VQ0J 16124774 IC50 = 86 nM T57700 CX7FV0 16124775 IC50 = 48 nM T57700 CGF2M4 16124831 IC50 = 42 nM T57700 C3FS0I 16124974 IC50 = 65 nM T57700 C3B8SQ 16124975 IC50 = 26 nM T57700 CD3U0I 16124976 IC50 = 32 nM T57700 C5W9ZT 16125110 IC50 = 11200 nM T57700 C9R4EN 16125232 IC50 = 17 nM T57700 C9XMJ4 16125233 IC50 = 10 nM T57700 CF23VU 16125380 IC50 = 10 nM T57700 CZM0J2 16125381 IC50 = 28 nM T57700 CVAZ06 16125453 IC50 = 61 nM T57700 CP3HS4 16220354 IC50 = 26 nM T57700 CDZ31W 16747696 IC50 = 49 nM T57700 CU35QY 16755735 IC50 = 250 nM T57700 CL9BQ6 17748275 IC50 = 17800 nM T57700 C25UKC 21081761 IC50 = 610 nM T57700 CGX61W 22041319 IC50 = 10 nM T57700 C3JWK1 23654166 IC50 = 110 nM T57700 CI6C1R 23658582 IC50 = 3 nM T57700 C2RV3U 24180608 IC50 > 30000 nM T57700 C3X1WH 24742411 IC50 = 4 nM T57700 CS78XJ 24742412 IC50 = 4 nM T57700 C2KA6G 24742584 IC50 = 3 nM T57700 CN9GC8 24742586 IC50 = 1 nM T57700 CA3I4T 24753787 IC50 > 50000 nM T57700 CY7FG8 24759282 IC50 = 2500 nM T57700 C9OM3V 24759285 IC50 = 1600 nM T57700 CWQR59 24759286 IC50 = 2400 nM T57700 C7YG1N 24759534 IC50 = 2700 nM T57700 CAJ4T2 24762205 IC50 = 89 nM T57700 CQNP54 24764449 IC50 = 10000 nM T57700 CCF17D 24768394 IC50 = 14800 nM T57700 CYK71D 24768395 IC50 > 12500 nM T57700 C7EXG0 24768396 IC50 > 12500 nM T57700 C0JUN4 24812717 IC50 = 6.1 nM T57700 CP6N9M 24812718 IC50 = 77 nM T57700 CW0G8H 24812719 IC50 = 28 nM T57700 CYBI02 24823426 IC50 = 5 nM T57700 CG0K1Z 24824046 IC50 = 14 nM T57700 CX0S9L 24854902 IC50 = 1174 nM T57700 C1SVT2 24854903 IC50 = 1061 nM T57700 C8DPJ4 24874843 IC50 = 250 nM T57700 CR5Z9A 24874845 IC50 = 1900 nM T57700 CPDY61 24874883 IC50 = 42 nM T57700 C25LQE 24874885 IC50 = 3000 nM T57700 CNHY40 24874886 IC50 = 510 nM T57700 CJ67CB 24874887 IC50 = 400 nM T57700 CJ0CK5 24875075 IC50 = 120 nM T57700 C5BLF1 24875123 IC50 = 890 nM T57700 C49KUH 24875222 IC50 = 300 nM T57700 C8A9FN 24875261 IC50 = 600 nM T57700 C85CSJ 24875262 IC50 = 40 nM T57700 CJ2CB0 24875263 IC50 = 57 nM T57700 C4BJK8 24875264 IC50 = 25 nM T57700 CE3IW4 24879184 IC50 = 14 nM T57700 C7V8BA 24879242 IC50 = 22 nM T57700 CT76XV 24879243 IC50 = 14 nM T57700 CGD8J5 24879244 IC50 = 17 nM T57700 C1XWO7 24879245 IC50 = 10 nM T57700 CA21RX 24879305 IC50 = 1 nM T57700 COF05N 24879306 IC50 = 210 nM T57700 C6NIQ2 24879307 IC50 = 2.1 nM T57700 C45HIT 24879308 IC50 = 7.9 nM T57700 CM6G7A 24879309 IC50 = 17 nM T57700 C0KW5Y 24879310 IC50 = 28 nM T57700 C7M9FB 24879311 IC50 = 40 nM T57700 C0ZJX6 24879366 IC50 = 20 nM T57700 C5NA4Z 24879367 IC50 = 13 nM T57700 CDJE41 24879368 IC50 = 16 nM T57700 C9B2TF 24880043 IC50 = 6 nM T57700 CFK2B9 24882503 IC50 = 930 nM T57700 C43HWQ 24883287 IC50 > 10000 nM T57700 C8DA5Q 24883334 IC50 > 10000 nM T57700 CY8L7E 24896769 IC50 > 10000 nM T57700 CIFO50 24897305 IC50 = 43 nM T57700 C5FD1A 24937369 IC50 = 6 nM T57700 C8DG1Y 24941253 IC50 = 2944 nM T57700 C15BZP 24949852 IC50 = 700 nM T57700 CZHE50 24949856 IC50 = 5900 nM T57700 CU7I2E 24963046 IC50 = 162 nM T57700 C9YN2Q 24967131 IC50 > 10000 nM T57700 C4EG8R 24993189 IC50 = 1904 nM T57700 C4KG0Y 25022599 IC50 = 170 nM T57700 C2ICS7 25065806 IC50 = 414 nM T57700 C35MEP 25068511 IC50 = 11 nM T57700 C5AQL3 25068516 IC50 = 11 nM T57700 CRM43Q 25068566 IC50 = 7 nM T57700 CN7H1J 25068567 IC50 = 28 nM T57700 CFJ6L3 25068568 IC50 = 170 nM T57700 C8TW5R 25068569 IC50 = 4 nM T57700 C7XWM4 25068620 IC50 = 1 nM T57700 CVT81X 25068621 IC50 = 2 nM T57700 C0MWF2 25068622 IC50 = 1 nM T57700 CPL3O0 25068623 IC50 = 3 nM T57700 C7EQ9F 25068624 IC50 = 4 nM T57700 CF73XJ 25068675 IC50 = 20 nM T57700 CKHU19 25069284 IC50 = 7 nM T57700 CBFU72 25069336 IC50 = 11 nM T57700 C0FB5J 25069338 IC50 = 5 nM T57700 CA48BZ 25069339 IC50 = 8 nM T57700 CRZF82 25069340 IC50 = 59 nM T57700 CH90KV 25097876 IC50 = 961 nM T57700 C9L5ID 25098154 IC50 > 1000 nM T57700 CAO38V 25098429 IC50 = 491 nM T57700 CQ27UI 25113814 IC50 = 4 nM T57700 C2IHY0 25114266 IC50 = 4 nM T57700 CP8S9W 25116064 IC50 = 8 nM T57700 CTV54O 25123227 IC50 = 150 nM T57700 C1IYN7 25127854 IC50 = 21 nM T57700 CKD14B 25127856 IC50 = 130 nM T57700 CJBX60 25128180 IC50 = 170 nM T57700 CC5SD9 25128181 IC50 = 240 nM T57700 CF7C5B 25129829 IC50 = 1061 nM T57700 CXNM84 25129830 IC50 = 529 nM T57700 CY2S1P 25129831 IC50 > 8331 nM T57700 C1NPM8 25130181 IC50 = 41 nM T57700 CL0Z1F 25181502 IC50 = 1600 nM T57700 C6FGQ1 25206346 IC50 = 430 nM T57700 CXNW87 25207322 IC50 = 1 nM T57700 CNG96H 25210579 IC50 > 10000 nM T57700 C2TXC6 25218656 IC50 = 13 nM T57700 CFU60Y 25235817 IC50 = 115 nM T57700 C8B6TY 42628503 EC50 < 500 nM T57700 CU9E4P 42629114 IC50 > 10000 nM T57700 CWT68J 44186427 IC50 = 21.9 nM T57700 CEL61X 44229839 IC50 > 10000 nM T57700 C0KD4U 44346053 IC50 > 10000 nM T57700 CYV2D7 44368815 IC50 = 105 nM T57700 C74BAO 44409484 IC50 = 623 nM T57700 C5OK1I 44409504 IC50 = 234 nM T57700 CS8YQ2 44414316 IC50 = 28 nM T57700 C7KZV2 44414322 IC50 = 103 nM T57700 CJM06T 44414347 IC50 = 145 nM T57700 CBZ2X3 44414348 IC50 = 69 nM T57700 C84DVH 44414371 IC50 > 50000 nM T57700 C32UEI 44414376 IC50 = 86 nM T57700 C45PBG 44414394 IC50 = 2190 nM T57700 CD1I5Y 44414395 IC50 > 50000 nM T57700 CF2JA5 44414419 IC50 = 75 nM T57700 C3G2FJ 44414460 IC50 = 101 nM T57700 C6YL5H 44414486 IC50 = 674 nM T57700 C5RTK0 44414527 IC50 = 17 nM T57700 CRL1C4 44414547 IC50 = 17239 nM T57700 C0MZ7P 44414549 IC50 = 36 nM T57700 C3SYD7 44414595 IC50 = 9746 nM T57700 CP6TZ2 44414596 IC50 = 4843 nM T57700 C6I8TW 44414597 IC50 = 19 nM T57700 CIQA35 44414621 IC50 = 136 nM T57700 CUW8C1 44414632 IC50 = 237 nM T57700 C06UCM 44414633 IC50 = 38 nM T57700 CQB17H 44414646 IC50 = 25 nM T57700 CLD07U 44414647 IC50 = 56 nM T57700 CTAZ73 44414648 IC50 = 59 nM T57700 C1XCW7 44414659 IC50 = 921 nM T57700 C1TR2Y 44414666 IC50 = 27 nM T57700 CBY7D9 44414679 IC50 = 18 nM T57700 CO14UX 44414683 IC50 = 1387 nM T57700 C1LZ9S 44414695 IC50 = 24 nM T57700 C0JF1Z 44414779 IC50 = 28 nM T57700 C0THE4 44414816 IC50 = 38 nM T57700 CRF01G 44414847 IC50 = 23829 nM T57700 CXV94N 44414848 IC50 = 139 nM T57700 CUI2N3 44414867 IC50 = 17 nM T57700 C8LH5Q 44414868 IC50 = 26845 nM T57700 CD13BL 44414880 IC50 = 13 nM T57700 CTCM71 44414881 IC50 = 5710 nM T57700 C51BYS 44420784 IC50 = 152 nM T57700 C5WGQ0 44421704 IC50 = 14735 nM T57700 CF34KY 44421705 IC50 = 96 nM T57700 CETQ79 44427518 IC50 = 31800 nM T57700 COPG94 44427519 IC50 > 10000 nM T57700 C14MTJ 44440231 IC50 > 50000 nM T57700 CA86YP 44440232 IC50 > 50000 nM T57700 COK21X 44440233 IC50 = 7180 nM T57700 CYMN10 44440242 IC50 = 5610 nM T57700 C96ARW 44440243 IC50 = 5150 nM T57700 CGL0R4 44440244 IC50 = 1670 nM T57700 CQI8S3 44440245 IC50 = 9540 nM T57700 CZM08I 44440246 IC50 = 1580 nM T57700 C4O8NF 44440247 IC50 = 2550 nM T57700 C1DAU0 44440248 IC50 = 4390 nM T57700 C93TBM 44440249 IC50 = 1120 nM T57700 C6VLC0 44440250 IC50 = 1100 nM T57700 CO37FE 44440251 IC50 = 900 nM T57700 C6T0IK 44440252 IC50 = 180 nM T57700 CJ05OC 44440253 IC50 = 4330 nM T57700 CGV37F 44440254 IC50 = 175 nM T57700 C5JUV3 44440256 IC50 = 4330 nM T57700 CFB56S 44440259 IC50 = 127 nM T57700 CEW9G2 44440261 IC50 = 619 nM T57700 CA5Q0P 44442388 IC50 = 2 nM T57700 C65YCN 44442389 IC50 = 58 nM T57700 CW02SD 44442390 IC50 = 42 nM T57700 C73GEP 44442391 IC50 = 45 nM T57700 CX56BF 44442392 IC50 = 17 nM T57700 C6L3GV 44442393 IC50 = 19 nM T57700 CX3J2I 44442394 IC50 = 18 nM T57700 C5QJ0P 44442395 IC50 = 1 nM T57700 CC3Z7Q 44442396 IC50 = 1 nM T57700 CLR10Z 44442397 IC50 = 37 nM T57700 C9UOK1 44442398 IC50 = 27 nM T57700 CE9T6W 44442399 IC50 = 72 nM T57700 CM6K2R 44442400 IC50 = 25 nM T57700 CW8JC5 44442401 IC50 = 50 nM T57700 CD1TY7 44442402 IC50 = 3 nM T57700 C4POG9 44442403 IC50 = 13 nM T57700 C0XHW1 44442404 IC50 = 8 nM T57700 CBSM51 44442405 IC50 = 12 nM T57700 CNT36H 44442406 IC50 = 9 nM T57700 CRA0Q8 44442407 IC50 = 4 nM T57700 C7YZ3M 44442408 IC50 = 20 nM T57700 CY9G0Q 44442409 IC50 = 23 nM T57700 C6XAR9 44442410 IC50 = 87 nM T57700 CJU4F6 44442411 IC50 = 240 nM T57700 CO0N1A 44442412 IC50 = 48 nM T57700 CIR9A7 44442413 IC50 = 12 nM T57700 CBQ51S 44442414 IC50 = 95 nM T57700 CHP41T 44442415 IC50 = 12 nM T57700 CI26UX 44442416 IC50 = 17 nM T57700 C2W1RN 44442417 IC50 = 4 nM T57700 C4A9FD 44442418 IC50 = 5 nM T57700 CKC3J0 44442419 IC50 = 19 nM T57700 C8W5YG 44447872 IC50 = 9 nM T57700 C13FIN 44450007 IC50 > 13000 nM T57700 CLK0W7 44453682 IC50 = 67 nM T57700 CF16QB 44560451 IC50 = 37 nM T57700 C0U8DH 44560546 IC50 = 108 nM T57700 CN3I8C 44560547 IC50 = 7 nM T57700 C0M1FW 44560587 IC50 = 58 nM T57700 C18JQN 44560588 IC50 = 2 nM T57700 C19KFW 44560589 IC50 = 120 nM T57700 C18WQN 44560590 IC50 = 4470 nM T57700 CS50FI 44560639 IC50 = 1180 nM T57700 CS8GY1 44560640 IC50 = 35 nM T57700 C6VF0N 44560641 IC50 = 9 nM T57700 C3QIX6 44560642 IC50 = 3640 nM T57700 C6I1TW 44560803 IC50 = 9 nM T57700 CXD9B4 44578561 IC50 = 3200 nM T57700 C9VXN3 44578709 IC50 > 10000 nM T57700 CY1A7W 44593407 IC50 = 18 nM T57700 CU3RF1 45139989 IC50 > 10000 nM T57700 CQGZ06 45139991 IC50 > 10000 nM T57700 CI82UE 45270897 IC50 > 5000 nM T57700 C4UM6Y 45273507 IC50 > 5000 nM T57700 C6E2SC 45482700 IC50 > 10000 nM T57700 CZXH74 45482750 IC50 > 10000 nM T57700 CA06GW 45487959 IC50 > 1000 nM T57700 CUMF37 45487992 IC50 > 1000 nM T57700 CFE79C 45487997 IC50 = 250 nM T57700 CNI92D 46182735 IC50 < 10 nM T57700 CUA97D 46209401 IC50 > 10000 nM T57700 CF57GK 46215462 IC50 = 1000 nM T57700 CY3HW5 46224684 IC50 > 10000 nM T57700 C2P9QO 46228508 IC50 = 1340 nM T57700 C6E5PY 46228822 IC50 = 883 nM T57700 C3T8AM 46228951 IC50 = 216 nM T57700 CYZV41 46231219 IC50 = 3467 nM T57700 C7J5UP 46231220 IC50 = 3330 nM T57700 CC96GZ 46231221 IC50 = 3219 nM T57700 CYT37A 46232443 IC50 = 41000 nM T57700 C48ZVW 46232555 IC50 > 50000 nM T57700 CS9B1U 46232556 IC50 = 41000 nM T57700 C7ON5A 46233287 IC50 > 10000 nM T57700 C9H4YO 46233889 IC50 = 610 nM T57700 CRT34L 46235770 IC50 = 20 nM T57700 CXFU08 46838910 IC50 = 6.8 nM T57700 C7NUY3 46847552 IC50 > 1000 nM T57700 CE3WH9 46865125 IC50 > 200000 nM T57700 C45LYT 46865445 IC50 > 200000 nM T57700 C1XEY4 46866615 IC50 > 200000 nM T57700 CF6K3E 46866616 IC50 > 200000 nM T57700 CQB16A 46872415 Ki > 4000 nM T57700 CLS29B 46872626 IC50 > 10000 nM T57700 C4DWZ6 46879153 IC50 = 200 nM T57700 C2O8RZ 46886323 IC50 > 1000 nM T57700 C0WYM1 46898022 IC50 = 1350 nM T57700 CTZ71Y 46898039 IC50 = 3.1 nM T57700 CQLT07 46913878 IC50 < 1000 nM T57700 C60GAV 46929544 IC50 = 1350 nM T57700 CC8FS1 49799031 IC50 = 1.5 nM T57700 C27SKR 49799067 IC50 = 14.4 nM T57700 CCX04I 49799068 IC50 = 9 nM T57700 CQZC18 49799069 IC50 = 16.2 nM T57700 C2HA1O 49799301 IC50 = 4.5 nM T57700 CZBW04 49799372 IC50 = 7.2 nM T57700 CHIQ50 49799374 IC50 = 6 nM T57700 C45FZO 49799375 IC50 = 3.3 nM T57700 C0SJ7Q 49804868 IC50 > 5000 nM T57700 CHSF07 49806372 IC50 > 1000 nM T57700 COR4V2 49806718 IC50 > 5000 nM T57700 C5ME3S 49806721 IC50 > 5000 nM T57700 C67HGW 49806722 IC50 = 1057 nM T57700 CY90BD 49818230 IC50 = 3000 nM T57700 CR58WT 49840391 IC50 = 1 nM T57700 CA2J6U 49840467 IC50 = 9 nM T57700 CB0S2P 49842666 IC50 = 1300 nM T57700 C5R6QY 49842669 IC50 > 100000 nM T57700 C0NA9U 49842670 IC50 = 2800 nM T57700 CC7MR2 49842671 IC50 = 47000 nM T57700 CAI20B 49842778 IC50 = 1300 nM T57700 CRA74I 49842779 IC50 = 4100 nM T57700 CF91RS 49843531 IC50 > 10000 nM T57700 CD3H8X 50925576 IC50 = 346 nM T57700 C2Y6QS 50938552 IC50 > 10000 nM T57700 CS9G6E 50997096 IC50 > 10000 nM T57700 C9NYP4 51036677 IC50 > 10000 nM T57700 C4WRY3 51037112 IC50 > 10000 nM T57700 CRI28Z 51037948 IC50 > 10000 nM T57700 CB9C8G 51351016 IC50 = 788 nM T57700 COD9Y2 51351017 IC50 = 788 nM T57700 CW96FU 51351018 IC50 = 4710 nM T57700 CR9T2E 51351019 IC50 = 2740 nM T57700 C1VML8 52936434 Ki = 12 nM T57700 CU1T5C 52936530 Ki = 12 nM T57700 CK69ML 52936531 Ki < 10 nM T57700 CCT6B9 52936532 Ki = 83 nM T57700 CC7SE4 52936533 Ki = 81 nM T57700 CA93FM 52936534 Ki = 155 nM T57700 C9KO7D 52936535 Ki = 270 nM T57700 CEQN27 52936621 Ki = 200 nM T57700 C2A6MX 52936622 Ki = 1300 nM T57700 CBH0K9 52936623 Ki = 400 nM T57700 CKF2D5 52936624 Ki = 400 nM T57700 CE6L8W 52950012 IC50 = 10.8 nM T57700 C7MC1H 52950013 IC50 = 125.8 nM T57700 C8ZTF9 53249002 IC50 = 2823 nM T57700 C09SDH 53257410 IC50 > 10000 nM T57700 C2P3OT 53316977 IC50 = 11000 nM T57700 CZ0BV7 53320342 IC50 = 7600 nM T57700 CX59LD 53320915 IC50 = 81000 nM T57700 CZY0J7 53323592 IC50 = 1400 nM T57700 C2W9OA 53324451 IC50 = 673 nM T57700 CCKD48 53324892 IC50 = 100000 nM T57700 CNPM14 53341082 IC50 > 3000 nM T57700 CM7P3W 53357328 IC50 > 50000 nM T57700 CBK9Q6 53357848 IC50 > 10000 nM T57700 C8NA4L 53384644 IC50 > 30000 nM T57700 CVG90B 53389651 IC50 > 10000 nM T57700 CKAP47 54578772 IC50 = 83.9 nM T57700 CR9F8Q 54578773 IC50 = 49.8 nM T57700 C4Z1NO 54578774 IC50 = 2422 nM T57700 CD6RH1 54578996 IC50 > 5000 nM T57700 CV79SW 54578997 IC50 > 5000 nM T57700 CO6B0E 54583043 IC50 > 10000 nM T57700 CY4O2I 54584313 IC50 = 2.1 nM T57700 C3PGE2 54585958 IC50 > 10000 nM T57700 CV7HJ8 54585959 IC50 > 10000 nM T57700 C0SC3J 54672928 IC50 = 80 nM T57700 CDMS75 54672929 IC50 = 40 nM T57700 CP5ZC3 54672931 IC50 = 89 nM T57700 C6OS4F 54672932 IC50 = 71 nM T57700 CR64QL 54673093 IC50 = 87 nM T57700 CE1D2H 54673094 IC50 = 98 nM T57700 CJL9T7 54673095 IC50 = 102 nM T57700 C73LSR 54673096 IC50 = 72 nM T57700 CE1ZK6 54759168 IC50 > 10000 nM T57700 C8AB1J 54759606 Ki = 200 nM T57700 C1XS2J 54760383 IC50 = 540 nM T57700 CBO2L1 54761157 IC50 = 7.9 nM T57700 CS23GM 54762055 IC50 = 8 nM T57700 CXQ0R1 56593680 Ki = 18 nM T57700 CSO49B 56593682 IC50 = 23 nM T57700 CUQ2Z3 56593684 Ki < 50 nM T57700 CVT2Y9 56593685 Ki = 21 nM T57700 C6VOK1 56593686 Ki = 10 nM T57700 CIMU73 56593834 Ki = 240 nM T57700 CCVD67 56593835 Ki = 180 nM T57700 CZIM93 56593836 Ki < 0.001 nM T57700 C6V9LJ 56593837 Ki < 50 nM T57700 CUP6Z9 56593838 Ki < 50 nM T57700 C5KR6N 56595558 Ki = 9 nM T57700 COI9U2 56595687 Ki = 12 nM T57700 CFY2I4 56595689 Ki = 60 nM T57700 CAM8E1 56595690 Ki = 37 nM T57700 C6ET0W 56595693 Ki = 270 nM T57700 CM8JX1 56604907 IC50 = 100 nM T57700 CQ17GA 56640518 IC50 > 200000 nM T57700 CG20VK 56640520 IC50 > 200000 nM T57700 CZ9C8M 56640588 IC50 > 200000 nM T57700 CH0D7P 56640590 IC50 > 200000 nM T57700 CFJ37O 56649380 IC50 = 77 nM T57700 CV8B1X 56649401 IC50 = 72 nM T57700 CUEW30 56649402 IC50 = 61 nM T57700 CK2OT6 56649403 IC50 = 83 nM T57700 CVN1Z8 56649405 IC50 = 96 nM T57700 CTR10F 56658543 Ki = 205 nM T57700 CJL83V 56682400 Ki < 50 nM T57700 CJBL48 56925034 IC50 = 41 nM T57700 C87YOZ 56929808 IC50 = 52 nM T57700 CY36EG 56945171 IC50 = 160 nM T57700 C4OG7H 56945172 IC50 = 720 nM T57700 CH0QA3 56945173 IC50 = 1100 nM T57700 CM0NQ5 56945174 IC50 = 2600 nM T57700 CXKF03 56945175 IC50 = 2300 nM T57700 C6WU4V 56945277 IC50 = 63 nM T57700 CP58NG 56954518 IC50 = 16 nM T57700 CI6QE5 56970263 IC50 < 500 nM T57700 C62OJE 56970264 IC50 = 600 nM T57700 C3UHX0 57394704 IC50 > 5000 nM T57700 C29ZPK 57395544 IC50 > 25000 nM T57700 CD7C4R 57396463 IC50 = 2991 nM T57700 CX2UW6 57399904 IC50 > 5000 nM T57700 CE31FR 57399905 IC50 > 5000 nM T57700 C3E4MA 57401677 IC50 > 5000 nM T57700 CP9Z4O 57403409 IC50 > 5000 nM T57700 CRU80Y 57403410 IC50 > 5000 nM T57700 CZSM95 57412684 IC50 = 6800 nM T57700 CE59QS 57505507 IC50 = 23 nM T57700 C8P6RD 57505528 IC50 = 120 nM T57700 CR1P7W 57598055 IC50 = 72.8 nM T57700 C4P8KD 57737398 IC50 = 230.7 nM T57700 C8R4FE 57991377 IC50 = 225.8 nM T57700 CVK0G4 58056356 IC50 > 50000 nM T57700 CH7L5N 58172700 IC50 < 10 nM T57700 CSP3L0 58994366 IC50 = 4000 nM T57700 CD2WR4 58994369 IC50 = 13 nM T57700 CK52WC 58994383 IC50 = 360 nM T57700 C9Q8AW 58994385 IC50 = 720 nM T57700 CX6K1H 58994468 IC50 = 6.1 nM T57700 C19ILC 58994517 IC50 = 110 nM T57700 C86KUI 58994523 IC50 = 100 nM T57700 CB8X9L 58994545 IC50 = 1900 nM T57700 C54MGH 58994552 IC50 = 250 nM T57700 CP6Q7F 58994591 IC50 = 1800 nM T57700 CK3LR6 58994593 IC50 = 530 nM T57700 C3L4JY 59176329 IC50 = 682 nM T57700 CZ3TG1 59375154 IC50 = 471 nM T57700 C4IBV1 59375998 IC50 = 1.4 nM T57700 CL3ND8 59376009 IC50 = 2.3 nM T57700 CC2AF9 59376012 IC50 = 5.8 nM T57700 CR7CG3 59376014 IC50 = 6.6 nM T57700 C60RIS 59376021 IC50 = 7.4 nM T57700 CT3Q5G 59376025 IC50 = 9.9 nM T57700 C97YSI 59376026 IC50 = 10.7 nM T57700 CEH5X6 59376027 IC50 = 2.1 nM T57700 C79EBT 59376032 IC50 = 7.8 nM T57700 C06DNI 59376037 IC50 = 2.7 nM T57700 C0XM7N 59376046 IC50 = 8.5 nM T57700 C70WCP 59376053 IC50 = 4.1 nM T57700 C5IHG9 59376058 IC50 = 5.7 nM T57700 CTK90V 59376059 IC50 = 180.8 nM T57700 C7ZY5I 59376061 IC50 = 35.5 nM T57700 CFT69X 59376062 IC50 = 255.7 nM T57700 C7D0BF 59376072 IC50 = 2 nM T57700 CD0RP7 59376074 IC50 = 43.1 nM T57700 C3HXC7 59376075 IC50 = 4.1 nM T57700 CAY6H8 59376079 IC50 = 6.9 nM T57700 CCX2W0 59376082 IC50 = 37.7 nM T57700 CXJ63M 59603829 IC50 = 810 nM T57700 CQEU96 59603842 IC50 = 690 nM T57700 CLH49Z 59790029 IC50 = 3 nM T57700 C1MR8Q 60097495 IC50 > 1000 nM T57700 C9QRX3 60098131 IC50 = 20 nM T57700 CQ4U2S 60154831 IC50 = 145 nM T57700 CKWI93 60155892 IC50 = 6.3 nM T57700 C3EK2G 60155994 IC50 = 63.8 nM T57700 CTR58Y 60199005 IC50 = 15 nM T57700 CA0LN1 60202314 IC50 = 2.7 nM T57700 CS1WL6 60202315 IC50 = 3.5 nM T57700 C7SGT6 60202316 IC50 = 3.3 nM T57700 C9ZCT2 62705065 IC50 > 1000 nM T57700 C51XCV 66781377 IC50 > 1000 nM T57700 C1HSE0 67035086 IC50 = 670 nM T57700 CWI6K5 67035106 IC50 > 10000 nM T57700 C38RGB 67035556 IC50 > 10000 nM T57700 CV63UL 67240318 IC50 > 10000 nM T57700 C8I7GC 68293638 IC50 > 10000 nM T57700 CD56XK 68293660 IC50 > 10000 nM T57700 CRH2Y9 68639605 IC50 = 756 nM T57700 C5DGR9 69036886 IC50 = 76 nM T57700 CH6S7Q 70681377 Ki = 39.81 nM T57700 CKY12U 70690667 Ki = 10 nM T57700 C6U8HO 70693451 IC50 = 27 nM T57700 CL4Z7S 70701950 IC50 = 7.6 nM T57700 CEBO91 71452977 IC50 > 10000 nM T57700 CAW17X 71494057 IC50 > 25000 nM T57700 CDE4X6 71494225 IC50 > 25000 nM T57700 CQY31T 71498139 IC50 = 3.9 nM T57700 C6HF8S 71521082 IC50 < 10 nM T57700 C9Z3AI 71521083 IC50 = 9.96 nM T57700 CCN01X 71547862 IC50 > 10000 nM T57700 C1IT5U 71550931 IC50 > 10000 nM T57700 CG1I5B 71550932 IC50 = 243 nM T57700 CDJY72 71568837 IC50 = 2800 nM T57700 CRX81Q 71575642 IC50 = 507 nM T57700 C8CAG7 71578921 IC50 > 10000 nM T57700 CZ31PU 71583657 IC50 > 10000 nM T57700 C1F5NV 71624671 IC50 = 67 nM T57700 CQE01I 71624672 IC50 = 16.7 nM T57700 CV8XI0 71624673 IC50 = 497 nM T57700 CY82NR 71624674 IC50 = 200 nM T57700 C0IM7Z 71624675 IC50 = 12.5 nM T57700 C6JS8P 71624676 IC50 = 457 nM T57700 C2F0QN 71624677 IC50 > 1000 nM T57700 CQ75IY 71624788 IC50 = 3.03 nM T57700 C6GT1Q 71624789 IC50 = 2.61 nM T57700 C6ZYR9 71624790 IC50 = 8320 nM T57700 CCSI30 71624792 IC50 = 29.6 nM T57700 C4JD7I 71624793 IC50 = 82.3 nM T57700 CS0AQ6 71624904 IC50 = 1.9 nM T57700 C23XIU 71624905 IC50 = 9.28 nM T57700 C4KTH9 71624906 IC50 = 99.5 nM T57700 C7BG9F 71624907 IC50 = 254 nM T57700 CC61DF 71624908 IC50 = 214 nM T57700 CRLN56 71624909 IC50 > 1000 nM T57700 CLO8V2 71625035 IC50 = 117 nM T57700 CQI0N1 71625036 IC50 = 18.8 nM T57700 CO41GB 71625037 IC50 = 82.4 nM T57700 CC68IJ 71625038 IC50 = 284 nM T57700 C4SV3X 71625039 IC50 = 257 nM T57700 CT2K6M 71625040 IC50 = 185 nM T57700 C6JZ2E 71625161 IC50 > 1000 nM T57700 CRGQ64 71625290 IC50 = 274 nM T57700 CP83JY 71625291 IC50 = 407 nM T57700 CGJ8H4 71625292 IC50 = 413 nM T57700 C0D4LN 71625406 IC50 > 1000 nM T57700 C9B1RV 71625407 IC50 > 1000 nM T57700 CKOL80 71625408 IC50 = 741 nM T57700 CQY4U2 71625409 IC50 = 1500 nM T57700 C1FAU8 71679855 IC50 = 230 nM T57700 C75QWC 71763641 IC50 = 69.3 nM T57700 CVJ7S2 71763642 IC50 = 7.3 nM T57700 C8M4HU 71763643 IC50 = 6.1 nM T57700 CM4X1R 71763869 IC50 = 20.9 nM T57700 CKN96V 71764058 IC50 = 9.2 nM T57700 C1K5HE 71764059 IC50 = 29.2 nM T57700 C42VJY 71764060 IC50 = 30.1 nM T57700 CWY6Z0 71764220 IC50 = 4.5 nM T57700 CUFY90 71764221 IC50 = 1 nM T57700 CD28XR 71816087 IC50 = 14 nM T57700 CCKL45 72191698 IC50 = 397.6 nM T57700 C60TUV 72737208 IC50 > 10000 nM T57700 CJ3WA6 72737404 IC50 > 10000 nM T57700 CIBU31 72792686 IC50 = 2.1 nM T57700 C6PQ5G 72792757 IC50 = 29.2 nM T57700 C8SIL6 73349435 IC50 = 449.7 nM T57700 C1V3NZ 73425588 IC50 = 8.18 nM T57700 C2PAK9 73438493 IC50 = 1509 nM T57700 C7M4FR 75201717 IC50 = 630 nM T57700 C0OJ7W 75201718 IC50 > 2000 nM T57700 C6S2ZO 75201851 IC50 > 2000 nM T57700 CBAT06 76071144 IC50 = 888 nM T57700 CH8W7D 77461036 IC50 > 1000 nM T57700 CA65HB 78319164 IC50 = 200 nM T57700 CCJ43A 86302281 IC50 > 10000 nM T57700 CPG3A5 86302574 IC50 > 30000 nM T57700 C08WGI 86566799 IC50 = 4.02 nM T57700 C2IP9D 86567333 IC50 = 5.8 nM T57700 CNR39Z 86763813 IC50 = 160 nM T57700 CR9V4A 86763924 IC50 = 310 nM T57700 CX94SV 86764031 IC50 = 140 nM T57700 CXW8T3 86764574 IC50 = 9.8 nM T57700 CTKA08 86764579 IC50 = 19 nM T57700 C31EBZ 88876355 IC50 = 97 nM T57700 C1HW4B 89735655 IC50 > 100000 nM T57700 CG5P9A 90153688 IC50 = 100 nM T57700 C5S3YB 90645165 IC50 = 4.32 nM T57700 CY0UC4 90645194 IC50 > 10000 nM T57700 CX29IY 90655145 IC50 > 10000 nM T57700 CJQ5N6 91936970 IC50 = 534000 nM T57700 C8F7XO 92131166 IC50 = 9.36 nM T57700 CS2J0P 101879051 IC50 = 128 nM T57700 C0R2OH 101879052 IC50 = 71 nM T57700 CK72FW 102129497 IC50 = 2.17 nM T57700 C5HRO7 102431711 IC50 = 7400 nM T57700 CTGP06 117996541 IC50 > 10000 nM T57700 C45RCJ 118072307 IC50 > 2000 nM T57700 CL0YO5 118443595 IC50 > 100 nM T57700 CDK5G4 118687517 IC50 = 6.9 nM T57700 CY7BI2 118706214 IC50 > 10000 nM T57700 CH2ZF1 118709500 IC50 = 29.2 nM T57700 C5BD7H 118709501 IC50 = 261.4 nM T57700 C1W4CV 118709542 IC50 = 520 nM T57700 C5SU1L 118709543 IC50 = 134.6 nM T57700 CU0TC5 118709544 IC50 = 32.1 nM T57700 CW5RO3 118709545 IC50 = 3330 nM T57700 C6EDP8 118709546 IC50 = 785 nM T57700 C3MJ0O 118709547 IC50 = 1330 nM T57700 C6OX7W 118709548 IC50 = 426 nM T57700 CANQ19 118709549 IC50 = 457 nM T57700 C4Z3ME 118709550 IC50 = 571.3 nM T57700 C0CLB5 118709551 IC50 = 32.1 nM T57700 CTS23O 118709552 IC50 = 102 nM T57700 C5O0IX 118709553 IC50 = 97.7 nM T57700 CUG48C 118709554 IC50 = 104 nM T57700 CB8J7X 118709555 IC50 = 1420 nM T57700 CA6G3X 118709556 IC50 > 10000 nM T57700 C6K5IJ 118709557 IC50 = 398 nM T57700 C0S2VK 118709558 IC50 = 670 nM T57700 C2O1PI 118709559 IC50 = 320 nM T57700 CXS09B 118709560 IC50 = 76.7 nM T57700 CWF87I 118709561 IC50 = 2260 nM T57700 CC8K3M 118709562 IC50 = 65.1 nM T57700 CDQ1X7 118709563 IC50 = 8.5 nM T57700 C1H3PL 118709564 IC50 = 8.8 nM T57700 C8HZA5 118709565 IC50 = 24.6 nM T57700 CE01TV 118709566 IC50 = 25.6 nM T57700 C9QPO2 118709567 IC50 = 10800 nM T57700 C8N4HO 118709568 IC50 = 9.1 nM T57700 CH81WR 118709569 IC50 = 67.8 nM T57700 C86MDP 118709570 IC50 = 26.2 nM T57700 CF9BE0 118709571 IC50 = 8540 nM T57700 CMOQ72 118709572 IC50 = 1520 nM T57700 C4AHL2 118711367 IC50 = 6100 nM T57700 CWO9B7 118715995 IC50 = 45 nM T57700 C46QUT 118717614 IC50 > 200000 nM T57700 CJC34Y 118717615 IC50 > 200000 nM T57700 CFEP93 118717616 IC50 > 200000 nM T57700 CEC4H0 118717617 IC50 > 200000 nM T57700 CU2TG3 118717618 IC50 > 200000 nM T57700 C5OL0W 118717619 IC50 > 200000 nM T57700 C3KLI5 118723185 IC50 = 900 nM T57700 CRQY80 118723194 IC50 = 2700 nM T57700 C7JYP8 118723210 IC50 = 2400 nM T57700 CI6QA2 118723212 IC50 = 400 nM T57700 C75PHN 119058124 IC50 > 10000 nM T57700 CKBP72 121231408 IC50 > 10000 nM T57700 C7QE2J 121513893 IC50 = 559 nM T57700 C81IFQ 122163152 IC50 > 100000 nM T57700 C08KEM 122179540 IC50 = 2200 nM T57700 C3AJ4C 122179546 IC50 = 5500 nM T57700 CG0RP7 122179547 IC50 = 790 nM T57700 C1A0SQ 122179548 IC50 = 7000 nM T57700 C42GSX 122180520 Ki > 4000 nM T57700 CN81HR 122181799 IC50 = 20 nM T57700 C8DJ3K 122181802 IC50 = 54 nM T57700 CWA94G 122182409 IC50 = 38.2 nM T57700 C49UGP 122187122 IC50 = 180 nM T57700 CFKD32 122191637 IC50 = 1050 nM T57700 C4X7SD 122192466 IC50 = 294 nM T57700 C1XHI4 122193762 IC50 = 3 nM T57700 CNX0Q2 122193763 IC50 = 1 nM T57700 CWV0C3 122193764 IC50 = 1 nM T57700 CSG98Y 122193765 IC50 = 6 nM T57700 CCLQ75 122193769 IC50 = 14 nM T57700 CXDR48 122193770 IC50 = 11 nM T57700 CPA8C5 122193773 IC50 = 17 nM T57700 CQL0W7 122197565 IC50 > 10000 nM T57700 CN41IF 122634050 IC50 > 10000 nM T57700 CD67LU 122705248 IC50 > 10000 nM T57700 CX63VW 122705258 IC50 > 10000 nM T57700 C76IKM 122705261 IC50 > 10000 nM T57700 CVH7Z1 123920373 IC50 = 4 nM T57700 C8ALO2 124088839 IC50 > 10000 nM T57700 C1XD6R 127029809 IC50 = 362.8 nM T57700 CI1E5W 127029864 IC50 = 324.58 nM T57700 CKS28E 127034802 IC50 > 1000 nM T57700 CC58IQ 127043948 IC50 = 99 nM T57700 CG8DA9 127045861 IC50 > 100000 nM T57700 CC4ND8 127046862 IC50 > 100000 nM T57700 CO25WH 127052538 IC50 > 10000 nM T57700 CF5D2Y 129318936 IC50 > 10000 nM T57700 CPFG86 130313537 IC50 = 0.12 nM T57700 C80JMK 130313548 IC50 = 71 nM T57700 C6RPF1 130364436 IC50 > 10000 nM T57700 CSY34O 130364443 IC50 > 10000 nM T57700 CI9H2W 130364450 IC50 > 10000 nM T57700 CM4TO5 130364451 IC50 > 10000 nM T57700 CV4DH7 130364460 IC50 > 10000 nM T57700 CW91ZV 130364461 IC50 > 10000 nM T57700 CQIZ43 130364463 IC50 > 10000 nM T57700 C4IKC6 130364464 IC50 > 10000 nM T57700 C0X6JS 130364465 IC50 > 10000 nM T57700 C0ZGC1 130364467 IC50 > 10000 nM T57700 CO9C5Q 130364468 IC50 > 10000 nM T57700 CQW3P1 130364471 IC50 > 10000 nM T57700 CHWX05 130364473 IC50 > 10000 nM T57700 CLB65Y 130364478 IC50 > 10000 nM T57700 CUZG19 130364481 IC50 > 10000 nM T57700 C34OMJ 130364482 IC50 > 10000 nM T57700 C6TWR3 130364484 IC50 > 10000 nM T57700 C8SF5Q 130364488 IC50 > 10000 nM T57700 CS5C4E 130364494 IC50 > 10000 nM T57700 CVQ32Y 130364503 IC50 > 10000 nM T57700 CV8B0Y 130364506 IC50 > 10000 nM T57700 CHX23J 130364524 IC50 > 10000 nM T57700 CHYL89 130364535 IC50 > 10000 nM T57700 C6OXE3 132134663 IC50 >= 1000 nM T57700 CUO0C5 132156633 IC50 > 10000 nM T57700 C6OMB1 132204257 IC50 = 83 nM T57700 C6SEM5 132520995 EC50 < 100 nM T57700 C6ROQ3 132546210 IC50 = 75 nM T57700 CJ04HZ 132585195 IC50 = 2.4 nM T57700 C53OJM 132607333 IC50 = 2.45 nM T57700 CMI3Q0 132819888 IC50 = 270 nM T57700 CERS64 132937256 IC50 > 30000 nM T57700 CB3SZ2 134135265 IC50 = 336 nM T57700 C32AGN 134136205 IC50 = 256 nM T57700 CN35SO 134146628 IC50 > 1000 nM T57700 CUKE45 134147919 IC50 = 3.38 nM T57700 CR4QC3 134152617 IC50 = 644 nM T57700 CGDL39 134155715 IC50 = 214 nM T57700 CQR94G 134198433 IC50 > 10000 nM T57700 CYL5V1 134694986 IC50 = 5396 nM T57700 CLCO61 135398510 IC50 = 1 nM T57700 CTJ48K 135524085 IC50 = 6100 nM T57700 CUT1W7 135524168 IC50 = 5200 nM T57700 CHA4N2 136013680 IC50 > 10 nM T57700 CJ7U4C 136053657 IC50 = 162.5 nM T57700 CG1R7B 136087060 IC50 = 5600 nM T57700 CS4R2M 136098630 IC50 = 7 nM T57700 CWM2S3 136098631 IC50 = 1107 nM T57700 CC52HL 136189674 IC50 > 3600 nM T57700 C9RE8D 136215817 IC50 = 652.5 nM T57700 C1YUD0 136219394 IC50 > 10 nM T57700 CIU8W3 136254389 IC50 > 10 nM T57700 CXC69T 137321158 IC50 = 182 nM T57700 CE75QD 137321162 IC50 = 64 nM T57700 C94NUE 137333440 IC50 = 60 nM T57700 C5PZ9U 137355929 IC50 = 100 nM T57700 C3Z7BX 137355931 IC50 = 56 nM T57700 CPF20O 137355933 IC50 > 1000 nM T57700 C37GOF 137355935 IC50 = 69 nM T57700 C9PVK0 137355939 IC50 = 53 nM T57700 C01WQT 137355941 IC50 = 123 nM T57700 CV9MO4 137355952 IC50 = 49 nM T57700 CWPA09 137355957 IC50 = 49 nM T57700 C8PFA4 137356361 IC50 = 47 nM T57700 C25ERN 137631967 IC50 > 10 nM T57700 CWO6X5 137632753 IC50 = 20 nM T57700 CH9MQ6 137632801 IC50 = 183.7 nM T57700 CE1B7Y 137633677 IC50 = 4794 nM T57700 CMY81W 137633944 IC50 = 7.2 nM T57700 CNX0F9 137634126 IC50 = 30 nM T57700 CHC70D 137634143 IC50 = 318.5 nM T57700 CPFH76 137634323 IC50 = 1416 nM T57700 CV6W3A 137634751 IC50 = 210 nM T57700 CS24ZE 137635122 IC50 = 1680 nM T57700 CILC91 137635352 IC50 = 2.6 nM T57700 CLU61E 137635383 IC50 = 900 nM T57700 CBP52G 137635849 IC50 = 3.7 nM T57700 CK8G2R 137636007 IC50 = 8.7 nM T57700 CZ3W9X 137636239 IC50 = 390 nM T57700 CEL8G1 137636465 IC50 = 3.5 nM T57700 C5VE4K 137636547 IC50 > 10000 nM T57700 CC1DK7 137636884 IC50 = 130 nM T57700 CL1Q8V 137637006 IC50 = 10890 nM T57700 C06JRX 137637094 IC50 > 10 nM T57700 C9H2CA 137637302 IC50 = 6.5 nM T57700 CLFR07 137637309 IC50 = 4581 nM T57700 CZ05TY 137637593 IC50 > 10000 nM T57700 CCF28G 137638542 IC50 = 100.3 nM T57700 C9IA2Q 137638780 IC50 = 2.6 nM T57700 CP2B8Y 137639044 IC50 = 21432 nM T57700 CI7WH5 137639132 IC50 = 26 nM T57700 C0SVI6 137639489 IC50 > 10000 nM T57700 C6GQ7X 137640210 IC50 > 10000 nM T57700 CI5K8B 137640242 IC50 = 20 nM T57700 CR30WV 137640970 IC50 = 116 nM T57700 CA70ZG 137641063 IC50 = 12 nM T57700 CW3C1G 137641107 IC50 = 3.9 nM T57700 CO05XC 137641159 IC50 = 3000 nM T57700 C0TOY1 137641923 IC50 = 6.2 nM T57700 CO18WK 137641971 IC50 = 144 nM T57700 C6HU2I 137642245 IC50 = 1039.3 nM T57700 CJ4S0F 137642960 IC50 = 1949 nM T57700 CVF3Y4 137643942 IC50 = 1831 nM T57700 C3X8JZ 137644493 IC50 > 10000 nM T57700 C9F6VM 137645016 IC50 = 20 nM T57700 C6PKY7 137645383 IC50 > 10000 nM T57700 C2BP8R 137645569 IC50 = 2.4 nM T57700 CF92BJ 137646079 IC50 = 397 nM T57700 CRM7F6 137646380 IC50 = 2147.2 nM T57700 CHOF26 137646593 IC50 = 180 nM T57700 C0XPI5 137646696 IC50 = 239.6 nM T57700 CDU7X6 137647023 IC50 = 7500 nM T57700 C5B7PN 137647552 IC50 = 9.3 nM T57700 CU3FK9 137647695 IC50 = 190 nM T57700 C0E5LD 137647791 IC50 = 20556 nM T57700 CB2S1Q 137647872 IC50 = 310 nM T57700 CITB67 137647879 IC50 = 6768 nM T57700 C8CYG9 137648008 IC50 = 120 nM T57700 CA0DL1 137648651 IC50 = 5900 nM T57700 CGI1F8 137649216 IC50 = 6.2 nM T57700 CTF9N6 137649662 IC50 = 1.4 nM T57700 C49LAY 137649772 IC50 = 3.3 nM T57700 CVK6O2 137650604 IC50 = 201 nM T57700 CME2B7 137651196 IC50 = 120.9 nM T57700 C1DK0P 137651391 IC50 > 10 nM T57700 CHR9E0 137651685 IC50 = 2500 nM T57700 CY53VO 137651787 IC50 > 10000 nM T57700 C3BU6H 137651848 IC50 = 2.1 nM T57700 CL2GW4 137652151 IC50 = 51 nM T57700 CEU20L 137652422 IC50 = 440 nM T57700 CHP3E8 137653224 IC50 = 78 nM T57700 CG3DS7 137653707 IC50 = 6.7 nM T57700 CZS0M4 137653919 IC50 = 1.9 nM T57700 C2BWK8 137654090 IC50 = 740 nM T57700 CS21QO 137654848 IC50 > 50000 nM T57700 CIS4O3 137655297 IC50 = 2402 nM T57700 C9ZIV1 137655363 IC50 = 12 nM T57700 C17LIA 137655641 IC50 = 227 nM T57700 CQ70VE 137655849 IC50 = 46064 nM T57700 CB3NC4 137656277 IC50 = 3.3 nM T57700 C3A0FZ 137656323 IC50 = 1.6 nM T57700 C0RQB3 137656341 IC50 = 553 nM T57700 CDU1V6 137656806 IC50 = 15000 nM T57700 CZ4C1M 137656917 IC50 = 14 nM T57700 C3QY0B 137657045 IC50 = 820 nM T57700 CO61JG 137657076 IC50 = 318 nM T57700 CF8VD5 137657326 IC50 = 2 nM T57700 CV9H6B 137657843 IC50 = 22056 nM T57700 CV5H3Z 137657932 IC50 > 10 nM T57700 C98AVI 137657952 IC50 > 50000 nM T57700 CPV1S9 137658287 IC50 = 279 nM T57700 C4AL3Z 137658384 IC50 = 555.7 nM T57700 CE8DW7 137658399 IC50 > 10000 nM T57700 C81LTC 137658404 IC50 = 19 nM T57700 CQMB10 137658515 IC50 = 2.1 nM T57700 CX53JP 137658925 IC50 = 320 nM T57700 CU61WM 137658936 IC50 > 10000 nM T57700 C4FKX3 137659066 IC50 = 2225 nM T57700 CKVU74 137659511 IC50 = 270 nM T57700 CKVS16 137659546 IC50 = 3.6 nM T57700 CM5T3L 137660584 IC50 = 38667 nM T57700 C7FZA8 137660733 IC50 = 6438 nM T57700 CCG6N4 137660759 IC50 = 1.9 nM T57700 C4U2GQ 137660913 IC50 = 2700 nM T57700 CD03NK 137661226 IC50 = 5970 nM T57700 C09NZL 137661683 IC50 = 3.7 nM T57700 CHB9P7 137661707 IC50 = 1.7 nM T57700 CIAT28 137661788 IC50 = 2.3 nM T57700 CY9N8Q 137662234 IC50 > 10000 nM T57700 CIWG23 138393067 IC50 = 125 nM T57700 CH6FJ1 138454786 IC50 > 300 nM T57700 CN0X5D 138454787 IC50 = 616 nM T57700 C07EKN 138454794 EC50 = 34 nM T57700 CM3A8O 139030333 IC50 = 8500 nM T57700 C6AK0N 139030518 IC50 = 8 nM T57700 CS9Z4A 141523058 IC50 > 50000 nM T57700 CUV1P6 141523059 IC50 > 50000 nM T57700 C2CZ1Q 141523061 IC50 > 50000 nM T57700 C98TNO 141523067 IC50 > 50000 nM T57700 CJQC54 141523068 IC50 > 50000 nM T57700 CW47GO 141523069 IC50 = 25800 nM T57700 CUV07Y 141523072 IC50 = 18600 nM T57700 CKBQ94 141523076 IC50 > 50000 nM T57700 C4ASE6 141523085 IC50 > 50000 nM T57700 CT37IP 141523091 IC50 > 50000 nM T57700 C4LA8F 141523094 IC50 = 49200 nM T57700 C34CKN 141523354 IC50 = 10.12 nM T57700 C4HB8M 145949394 IC50 = 29 nM T57700 CB3Z1W 145949428 IC50 = 68.9 nM T57700 C0V8SM 145954139 IC50 = 10 nM T57700 C5VSC7 145956704 IC50 = 13400 nM T57700 CJT41L 145962084 IC50 = 2200 nM T57700 C65YWX 145964882 IC50 = 1800 nM T57700 CHC3T0 145965031 IC50 > 10000 nM T57700 CP92ZF 145965329 IC50 = 1100 nM T57700 C9HXI4 145966620 IC50 > 10000 nM T57700 CTUF34 145966712 IC50 = 163 nM T57700 CQE9M5 145966810 IC50 = 360 nM T57700 C1EH6C 145967078 IC50 > 10000 nM T57700 CDW83M 145967332 IC50 = 258.7 nM T57700 C5E8ZK 145968310 IC50 = 701 nM T57700 CHAU61 145968737 IC50 = 535 nM T57700 CWJ12M 145969155 IC50 = 68 nM T57700 CGW5S1 145969844 IC50 > 10000 nM T57700 CB8R3A 145970271 IC50 > 10000 nM T57700 C8NK3O 145970839 IC50 > 1000 nM T57700 C40VIL 145972979 IC50 = 7500 nM T57700 CQBY19 145974023 IC50 > 10000 nM T57700 CXRY95 145974888 IC50 = 3700 nM T57700 C74TYP 145975351 IC50 = 529.3 nM T57700 C4X7CT 145977420 IC50 > 10000 nM T57700 CLA57T 145978300 IC50 > 10000 nM T57700 CUNA14 145983151 IC50 > 50000 nM T57700 CD39VL 145983968 IC50 = 31300 nM T57700 C3L9WK 145984021 IC50 > 50000 nM T57700 C1Y5MO 145987062 IC50 = 684.5 nM T57700 CI85EU 145998085 IC50 = 3438 nM T57700 CD49VM 155295006 IC50 > 10000 nM T57700 CSHC63 155510467 IC50 > 10000 nM T57700 CG09WO 155512858 IC50 > 10000 nM T57700 C6H8ZU 155513172 IC50 = 2917 nM T57700 C2MD1Q 155513187 IC50 > 10000 nM T57700 C91EIC 155513236 IC50 = 950 nM T57700 CZDH58 155514096 IC50 > 10000 nM T57700 CZ0RI7 155517469 IC50 = 830 nM T57700 C84GJO 155517474 IC50 = 8414 nM T57700 C86HPW 155518524 IC50 = 11000 nM T57700 C63PZX 155518871 IC50 > 10000 nM T57700 C3VTM7 155519139 IC50 = 352 nM T57700 CM51TE 155519497 IC50 = 29 nM T57700 CU6Z5O 155520650 IC50 = 250 nM T57700 CN8F2P 155521009 IC50 = 82 nM T57700 CHP7Q9 155521761 IC50 = 100 nM T57700 CZ6XM2 155526493 IC50 = 122 nM T57700 CNP8T7 155530083 IC50 = 72.4 nM T57700 C0N7SQ 155531512 IC50 = 43 nM T57700 CK10UA 155531677 IC50 = 4994 nM T57700 CWLZ25 155535008 IC50 > 10000 nM T57700 CHOC87 155535920 IC50 > 2000 nM T57700 C8H1CZ 155536201 IC50 = 8300 nM T57700 C8NA6L 155536370 IC50 = 619.7 nM T57700 C9NX0I 155536511 IC50 = 130 nM T57700 C3LC9I 155536820 IC50 = 47.39 nM T57700 C0U3RI 155539733 IC50 = 24 nM T57700 C3Q9UA 155541932 IC50 = 1686 nM T57700 CWK26R 155544890 IC50 = 98 nM T57700 CYM14Z 155545786 IC50 = 86 nM T57700 CC9LQ2 155546287 IC50 > 20000 nM T57700 C2Z3PX 155546437 IC50 > 2000 nM T57700 CI27QV 155546853 IC50 > 10000 nM T57700 C7SF2C 155547229 IC50 = 380 nM T57700 CYP2O5 155547984 IC50 > 10000 nM T57700 C52UAJ 155551442 IC50 > 2000 nM T57700 CL8KR2 155552517 IC50 = 4934 nM T57700 CQ92ZH 155552526 IC50 = 91 nM T57700 C1TA9J 155553503 IC50 > 10000 nM T57700 C1WNS6 155553519 IC50 = 50 nM T57700 CN2WU7 155553601 IC50 = 38 nM T57700 C8BAU3 155554243 IC50 > 10000 nM T57700 CCQF25 155555943 IC50 > 10000 nM T57700 CHLY93 155562871 IC50 = 6591 nM T57700 C81JZW 155563388 IC50 = 5160 nM T57700 C60KLJ 155564326 IC50 = 3984 nM T57700 C4BS6J 155565938 IC50 = 3721 nM T57700 CINX89 155566065 IC50 = 8990 nM T57700 C7Q4RY 155566792 IC50 = 5978 nM T57700 C85WEG 155567932 IC50 = 107 nM T57700 CP69SU 155567937 IC50 > 10000 nM T57700 D00DNY 3213 IC50 = 200 nM T57700 D00ERW 44444843 Ki = 1119 nM T57700 D00HVA 11624601 Ki > 1200 nM T57700 D02BXJ 46864270 IC50 > 3000 nM T57700 D02RWC 59397065 IC50 = 1000 nM T57700 D03DZO 11715767 IC50 > 10000 nM T57700 D05FFB 91643 IC50 = 10 nM T57700 D05MHL 44605611 Ki = 190 nM T57700 D06HVH 54613583 IC50 > 10000 nM T57700 D07SRX 9797919 IC50 = 240 nM T57700 D08HFG 24809764 IC50 > 10000 nM T57700 D08ZWJ 97080 IC50 = 200 nM T57700 D09HVH 135566652 IC50 > 10 nM T57700 D09LPL 5329103 IC50 = 10 nM T57700 D09TNR 9850161 IC50 = 69 nM T57700 D0BL0O 71624791 IC50 = 4.89 nM T57700 D0BW4G 10907042 IC50 = 50 nM T57700 D0C2GE 67161540 IC50 = 11 nM T57700 D0CM6T 11314340 Ki = 5800 nM T57700 D0D6MH 11617559 IC50 > 13000 nM T57700 D0EE6A 6398883 IC50 = 236 nM T57700 D0GW4Q 5330524 IC50 = 290 nM T57700 D0I3XZ 11601743 IC50 = 500 nM T57700 D0L3JR 25212148 IC50 = 6 nM T57700 D0M4QA 56935577 IC50 = 5 nM T57700 D0N4LR 53469448 IC50 = 154 nM T57700 D0OZ2S 11785878 IC50 = 560 nM T57700 D0P3JW 447700 IC50 = 636 nM T57700 D0Q3NG 11715520 Ki > 1200 nM T57700 D0Q4EQ 16742063 IC50 = 513 nM T57700 D0R2WK 16038120 EC50 > 1000 nM T57700 D0S7IE 11658882 Ki > 1200 nM T57700 D0T4SL 72512 IC50 = 300 nM T57700 D0T8NU 16757525 IC50 > 4000 nM T57700 D0U3WQ 9817165 IC50 = 1000 nM T57700 D0UN9O 3385203 IC50 = 300 nM T57700 D0V4EX 54760053 IC50 = 1.2 nM T57700 D0X6KS 16125109 IC50 = 12500 nM T57700 D0Y4BL 11676971 IC50 = 5 nM T57700 D0Y9GK 16125106 IC50 = 7360 nM T74166 D05QNO 2968 IC50 ~ 1700 nM T74166 D0K0KH 656665 IC50 = 1800 nM T74166 D0K7WK 4595 IC50 = 27000 nM T74166 D0LM4A 170361 Ki = 74.7 nM T74166 D0Q9HF 187 EC50 = 19000 nM T74166 D0T8GD 89594 Ki = 260 nM T74166 D0V8HA 4032 IC50 = 100 nM T74166 D0X4ZR 444 IC50 = 1.8 nM T74166 D00EZO 10176607 Ki = 1200 nM T74166 D05RSC 10131048 EC50 = 1445.44 nM T74166 D08XPW 10235 Ki = 280 nM T74166 D0Y6OE 5310969 EC50 = 700 nM T74166 D0ZC3C 5310985 Ki = 2500 nM T74166 D03UID 5310967 Ki = 5400 nM T74166 D04HYP 3075702 EC50 = 190 nM T74166 D06LKM 11243536 IC50 >= 60000 nM T74166 D09ADT 119380 EC50 = 64000 nM T74166 D0A5RD 9795056 IC50 = 3300 nM T74166 D0AB4Q 9824145 EC50 > 10000 nM T74166 D0C9KD 44327552 Ki = 0.527 nM T74166 D0Y9HH 3036156 EC50 = 10000 nM T74166 C48GPY 5475 EC50 > 10000 nM T74166 C1O2ZJ 6059 IC50 ~ 1700 nM T74166 C5H9CN 9287 Ki > 10000 nM T74166 C4WTQ3 18985 Ki = 107 nM T74166 C2NM4A 72503 IC50 = 48200 nM T74166 CC3OR4 133106 EC50 = 34000 nM T74166 C2JM5W 202718 IC50 = 380.19 nM T74166 CK6SL0 666124 IC50 > 100000 nM T74166 CN6V5X 852545 Ki = 8500 nM T74166 C03FIQ 902985 IC50 = 17400 nM T74166 CF42DT 1094969 IC50 = 29600 nM T74166 CR2T7N 1302023 IC50 = 11600 nM T74166 CS1DC9 1307388 IC50 = 7600 nM T74166 C6C7UX 2268445 IC50 = 61400 nM T74166 CIN1G2 2655600 IC50 = 4000 nM T74166 CHX06D 2995464 IC50 = 31700 nM T74166 C3XM0R 3241687 IC50 = 19600 nM T74166 CAM0K9 3464560 IC50 = 15400 nM T74166 C9N6GB 3480598 IC50 = 17100 nM T74166 C9O7SE 3691150 IC50 = 99800 nM T74166 CHE9U8 4546524 IC50 = 11100 nM T74166 CRC58X 4779153 IC50 = 18200 nM T74166 C1EVM7 5310971 IC50 > 1000000 nM T74166 C5FQ4L 5364095 Ki = 2100 nM T74166 CF1NW5 6456944 IC50 = 46300 nM T74166 C69QWU 6471751 IC50 = 24700 nM T74166 C7M3WF 6472114 IC50 = 21700 nM T74166 CJ3FS9 6603935 IC50 = 50 nM T74166 CLM7T3 6918622 IC50 = 8800 nM T74166 CUN02J 7582345 IC50 > 100000 nM T74166 C81GRQ 8747436 IC50 = 18500 nM T74166 C50RLZ 8749430 IC50 = 19100 nM T74166 CZ69HA 9104895 IC50 = 16400 nM T74166 C08MRI 9794019 Ki = 1190 nM T74166 CKI6W9 9794220 Ki = 1600 nM T74166 C6YDQ0 9795278 Ki >= 60000 nM T74166 C2SHJ3 9812995 EC50 = 1540 nM T74166 C9YE1X 9813282 EC50 = 600 nM T74166 C9R8VP 9813576 EC50 = 2600 nM T74166 C27UWZ 9813730 EC50 = 3090.3 nM T74166 CFLI74 9813803 EC50 = 4073.8 nM T74166 C1M0SN 9815622 Ki = 810 nM T74166 CG4JD8 9815827 Ki = 4.9 nM T74166 CAT7Z4 9816191 Ki = 210 nM T74166 C71JPQ 9822806 IC50 = 9200 nM T74166 C5OL1T 9834096 EC50 = 9700 nM T74166 CHDY16 9834184 Ki = 710 nM T74166 C6FXS4 9834228 EC50 = 13182.57 nM T74166 C65DLA 9834234 EC50 = 12302.69 nM T74166 C80NVH 9834302 Ki = 810 nM T74166 C2D4HG 9834307 EC50 = 1200 nM T74166 CO9DY5 9834308 EC50 = 1100 nM T74166 CQY34E 9834353 EC50 = 5560 nM T74166 CQ98AW 9834452 EC50 = 25 nM T74166 CUB3G9 9834620 EC50 = 295.12 nM T74166 C95UWI 9837971 EC50 = 6400 nM T74166 CJ7CI4 9855608 EC50 = 2940 nM T74166 C4MG8D 9855694 EC50 = 1698.24 nM T74166 CBSF19 9855936 EC50 = 4360 nM T74166 CZS71O 9855966 EC50 = 2187.76 nM T74166 C10LFH 9856458 EC50 = 338.84 nM T74166 CZB45J 9856887 EC50 = 1949.84 nM T74166 CB6Z8S 9877653 EC50 = 77624.71 nM T74166 CSP4D2 9877707 EC50 = 25118.86 nM T74166 CFO4D6 9877782 EC50 = 2560 nM T74166 C7LD1U 9899354 EC50 = 1380.38 nM T74166 CRST76 9899814 Ki = 240 nM T74166 CX73LN 9917490 IC50 = 6800 nM T74166 CAJ1X8 9920686 Ki = 6.6 nM T74166 CTE89G 9921869 EC50 = 1800 nM T74166 C0C7NV 9930121 IC50 > 100000 nM T74166 CAV98S 9942481 EC50 = 30902.95 nM T74166 CVYM29 9942613 EC50 = 63095.73 nM T74166 C8ETL1 9942787 EC50 = 1905.46 nM T74166 COD73F 9943346 IC50 > 100000 nM T74166 C6AZ3X 9943908 IC50 = 11000 nM T74166 CY2Q8J 9964230 EC50 = 6100 nM T74166 CZE08N 9964805 EC50 = 1000 nM T74166 CGH81K 10051792 IC50 = 1200 nM T74166 C6XFH7 10058322 EC50 = 47.86 nM T74166 CGM3W9 10059716 Ki = 560 nM T74166 CJ6B2U 10081505 EC50 = 300 nM T74166 COE53P 10082341 EC50 = 28.84 nM T74166 CUW85L 10085732 EC50 > 100000 nM T74166 CCZ3T9 10130346 Ki = 1000 nM T74166 CTV58J 10130408 Ki = 69 nM T74166 C63VHC 10154344 Ki = 122 nM T74166 C1X0LJ 10176791 Ki = 980 nM T74166 C5WS0X 10198058 Ki = 2850 nM T74166 CBS1I4 10219939 Ki = 0.944 nM T74166 CN2JQ8 10262309 EC50 > 100000 nM T74166 CX8B5S 10267729 EC50 > 10000 nM T74166 C5AN1L 10375812 EC50 = 400 nM T74166 CLC49H 10421899 Ki = 1100 nM T74166 CRNE59 10443009 Ki = 3600 nM T74166 CNY59C 10443079 EC50 = 34.67 nM T74166 CHR72Q 10443815 Ki = 2400 nM T74166 CLDM93 10445840 IC50 = 81000 nM T74166 C8BCV0 10465833 EC50 = 1000 nM T74166 C64WPE 10559473 EC50 = 7000 nM T74166 C5PNA6 10799794 Ki = 946 nM T74166 CN0JI4 10911949 IC50 > 100000 nM T74166 CZR3T6 10932563 IC50 = 91 nM T74166 CG2D7O 11096168 Ki = 749 nM T74166 CLD5Z0 11098414 IC50 = 400 nM T74166 C5EO2P 11151120 EC50 = 13800 nM T74166 CMH15U 11201533 EC50 > 1000000 nM T74166 CJ3H1Q 11211996 EC50 > 1000000 nM T74166 C0F8MZ 11258762 EC50 = 18240 nM T74166 CW7JD6 11393999 EC50 = 26360 nM T74166 CU1S6Y 11400044 IC50 = 0.93 nM T74166 CJ61TB 11403803 EC50 = 20810 nM T74166 C57YWO 11422871 IC50 = 1.74 nM T74166 C5JT1E 11425617 EC50 > 1000000 nM T74166 CP1WH5 11461365 EC50 > 100000 nM T74166 CT1XJ7 11528487 EC50 > 100000 nM T74166 CYG3H9 11543786 IC50 = 38000 nM T74166 CBT1K9 11672813 Ki > 500 nM T74166 CN4Z5C 11679149 IC50 = 19952.62 nM T74166 C91PVY 11708150 Ki > 500 nM T74166 CA1C9Y 11715647 EC50 > 100000 nM T74166 CL15NV 11829725 Ki = 194 nM T74166 C8AN1M 12009050 Ki = 108 nM T74166 CF96QD 12303261 IC50 = 2620 nM T74166 CLJ14R 12358972 IC50 = 200 nM T74166 C0IJV5 12392828 IC50 = 10700 nM T74166 CE5X1A 12625600 Ki = 370 nM T74166 C3IV5B 14806309 IC50 = 0.46 nM T74166 C8T0DI 15519735 IC50 = 15.6 nM T74166 C7LF3K 16099069 EC50 = 257.04 nM T74166 CJLU49 16099070 EC50 = 950 nM T74166 CJH4F0 16099071 EC50 = 9.9 nM T74166 C52LBH 16099072 EC50 = 8.128 nM T74166 CXN75R 16099073 EC50 = 7.2 nM T74166 CGU63X 16099074 EC50 = 180 nM T74166 C4FEW3 16099075 EC50 = 1096.48 nM T74166 C6OR8V 16099076 EC50 = 2398.83 nM T74166 C91AUD 16099077 EC50 = 2800 nM T74166 C21YIA 16099078 EC50 = 389.05 nM T74166 CXD7Z3 16099079 EC50 = 7.943 nM T74166 C0WZR4 16099080 EC50 = 4.365 nM T74166 CLR21F 16099081 EC50 = 2951.21 nM T74166 CQ0C2P 16099082 EC50 = 238 nM T74166 CUI8P1 16099083 EC50 = 7413.1 nM T74166 C9PRA2 16099084 EC50 = 108 nM T74166 CI5K4R 16099085 EC50 = 64.8 nM T74166 C0GV4U 16099091 EC50 = 109.65 nM T74166 C83HRV 16099099 EC50 = 75.86 nM T74166 CFV86M 16099100 EC50 = 109.65 nM T74166 CVN2J3 16099101 EC50 = 70.79 nM T74166 CC9DA0 16099102 EC50 = 489.78 nM T74166 CQS1C4 16099103 EC50 = 4466.84 nM T74166 CDQF19 16099104 EC50 = 123.03 nM T74166 C3K8CO 16099105 EC50 = 1400 nM T74166 CWB4P7 16099106 EC50 = 830 nM T74166 CJ1P6E 16099107 EC50 = 158.49 nM T74166 CM9G0S 16099108 EC50 = 5700 nM T74166 CU5J2I 16099109 EC50 = 1513.56 nM T74166 C7S1GW 16099110 EC50 = 202 nM T74166 CZB59V 16099111 EC50 = 794 nM T74166 CZ94VM 16099112 EC50 = 23300 nM T74166 C2EIJ5 16099113 EC50 = 9940 nM T74166 CL5CR3 16099114 EC50 = 1020 nM T74166 C9XZI4 16099115 EC50 = 394 nM T74166 CO8ID2 16126643 Ki = 1200 nM T74166 CGZN70 16637618 Ki = 385 nM T74166 CHT0S5 17384430 IC50 > 100000 nM T74166 C1OTB6 18177037 EC50 = 28000 nM T74166 C3XHW0 18180401 EC50 > 10000 nM T74166 CXQM78 20695745 IC50 = 1.2 nM T74166 C4PJN6 21574409 Ki = 9.51 nM T74166 C0EO2W 22215312 Ki = 2450 nM T74166 C6EX4B 22291236 EC50 > 100000 nM T74166 C4OL6R 23169640 IC50 = 398.11 nM T74166 CVUW34 23251657 Ki = 37000 nM T74166 CXWI74 23332842 EC50 > 100000 nM T74166 CBQS32 23634540 EC50 = 1000 nM T74166 CI4GY6 23634543 EC50 = 3235.94 nM T74166 CZC61E 23634545 EC50 = 900 nM T74166 C2P6RE 23634548 EC50 = 87.1 nM T74166 C59MUH 23634670 EC50 = 177.83 nM T74166 CJY49C 23634788 EC50 = 8000 nM T74166 CBS3A5 23634911 EC50 = 1096.48 nM T74166 CSYC96 23634914 EC50 = 20892.96 nM T74166 C4CR5U 23634916 EC50 = 1258.93 nM T74166 CQUI19 23635035 EC50 = 588.84 nM T74166 C2GAQ9 23635037 EC50 = 3981.07 nM T74166 CUB17S 23635157 EC50 = 676.08 nM T74166 CM19ZP 23635159 EC50 = 16900 nM T74166 C1H7CZ 23635160 EC50 = 6025.6 nM T74166 CIK9U8 23635162 EC50 = 3235.94 nM T74166 C5KOC7 23635288 EC50 = 575.44 nM T74166 C15KIQ 23635417 EC50 = 22908.68 nM T74166 CVD51I 23635423 EC50 = 12022.64 nM T74166 CD94YA 23635530 EC50 = 2089.3 nM T74166 CCJ24W 23635651 EC50 = 602.56 nM T74166 CRE52L 23635654 EC50 = 9100 nM T74166 CI8VQ9 23635786 EC50 = 46773.51 nM T74166 CX52UA 23636037 EC50 = 50 nM T74166 CG2D4Y 23636156 EC50 = 4168.69 nM T74166 C2X7UR 23636160 EC50 = 1584.89 nM T74166 CB18JU 23636165 EC50 = 100 nM T74166 CMI29X 23636510 EC50 = 200 nM T74166 CDKB19 23636512 EC50 = 25118.86 nM T74166 C2JG3M 23636514 EC50 = 7079.46 nM T74166 C3QEI4 24686533 IC50 = 17500 nM T74166 CE2XP4 24795080 Ki > 10000 nM T74166 C84AQE 24945028 EC50 = 42000 nM T74166 CHY7C1 24945029 Ki = 2200 nM T74166 CV07CE 24945030 Ki > 10000 nM T74166 C30XMU 24945031 Ki = 2400 nM T74166 CGI46H 24945032 Ki = 3800 nM T74166 C50QZG 24945033 Ki = 7200 nM T74166 CT13LF 24945123 Ki = 4800 nM T74166 CI0YH2 24945124 EC50 = 79000 nM T74166 C3WIQ9 24945126 Ki = 11000 nM T74166 C93SUY 24945129 Ki = 7100 nM T74166 C5MNT9 24945296 Ki = 5400 nM T74166 C78HXO 24945297 Ki = 8100 nM T74166 CY5D6P 24945298 Ki > 10000 nM T74166 C1T0FO 24945299 Ki > 10000 nM T74166 C3UP8T 24945300 Ki = 8700 nM T74166 CKJG57 24945301 Ki = 6400 nM T74166 CW9F1R 24945302 Ki = 6500 nM T74166 C0N7YV 24945376 Ki = 6500 nM T74166 C3LBH5 24945542 Ki > 10000 nM T74166 CRYT93 24970319 Ki = 400 nM T74166 CD2CK3 25085910 IC50 = 167000 nM T74166 CT8N7H 25194896 Ki = 8200 nM T74166 C06EBO 27185027 IC50 = 11200 nM T74166 CY1I9X 29354120 IC50 = 13600 nM T74166 CGKR74 37066353 IC50 = 49600 nM T74166 C0DJ8H 39010244 IC50 = 95000 nM T74166 C1CWU0 42631007 IC50 = 1258.93 nM T74166 CJV6A7 44158944 IC50 = 800 nM T74166 C6NT5U 44190553 Ki = 4700 nM T74166 C6TOC5 44199430 Ki = 2100 nM T74166 C43GIX 44222896 EC50 = 5900 nM T74166 CBP9G1 44222951 Ki = 110 nM T74166 CN9CA4 44223026 Ki = 14000 nM T74166 C6MCF2 44223074 Ki = 670 nM T74166 CG5Q6P 44223132 Ki = 5500 nM T74166 CNP36F 44224169 EC50 = 6900 nM T74166 C4W0SH 44247585 EC50 > 100000 nM T74166 CH1OX8 44313307 Ki = 4500 nM T74166 CTMR48 44324442 Ki = 88 nM T74166 C5R4WQ 44348072 IC50 = 4265.8 nM T74166 CH7F9J 44348080 IC50 = 5200 nM T74166 CE6U1G 44348090 IC50 = 3200 nM T74166 C6OJD1 44348101 IC50 = 1700 nM T74166 CYW90O 44348287 IC50 = 1500 nM T74166 CSD9M7 44348293 IC50 = 2500 nM T74166 C8RAO6 44348296 IC50 = 1700 nM T74166 COA40Y 44348309 IC50 = 5888.44 nM T74166 CR42HE 44348319 IC50 = 3000 nM T74166 CZ2C4O 44348367 IC50 = 1300 nM T74166 CQ32NT 44348375 IC50 = 4500 nM T74166 C4XKW0 44348376 IC50 = 5011.87 nM T74166 C0SOG1 44348388 IC50 = 3200 nM T74166 CVGZ81 44348389 IC50 = 22908.68 nM T74166 CE8Z5V 44348411 IC50 = 1300 nM T74166 C1XEL6 44348526 IC50 = 6000 nM T74166 CRC25U 44354684 IC50 = 43000 nM T74166 CH3VS0 44395275 Ki = 2.35 nM T74166 C75SYG 44398004 IC50 > 750 nM T74166 C5L7UK 44398089 IC50 = 200 nM T74166 C1C3EN 44398092 IC50 = 1.5 nM T74166 C0LN4Z 44398101 IC50 > 750 nM T74166 C2K1WB 44398115 IC50 = 730 nM T74166 C52SCF 44398143 IC50 = 1 nM T74166 CYOE97 44399319 Ki = 1900 nM T74166 CN37JP 44419364 Ki = 0.16 nM T74166 C0BN3A 44421466 EC50 > 1000000 nM T74166 C5Q3NI 44542504 IC50 = 3.3 nM T74166 CYX7H5 44542510 IC50 = 0.65 nM T74166 C71QGD 44542511 IC50 = 3.1 nM T74166 C2EDU6 44542955 IC50 = 10 nM T74166 C03MXJ 44543264 IC50 = 2.6 nM T74166 CL5UK7 44543265 IC50 = 2.9 nM T74166 CM8U6J 44570006 Ki = 12589.25 nM T74166 CH84MQ 44570007 Ki = 25000 nM T74166 C2E3LJ 44570008 Ki = 1400 nM T74166 CWPR65 44570009 Ki = 3162.28 nM T74166 C13RLY 44570010 Ki = 12000 nM T74166 CIV69B 44570011 Ki = 4900 nM T74166 CG4YE9 44570012 Ki = 1995.26 nM T74166 C0ZL8N 44570053 EC50 = 1000 nM T74166 CQ4K3T 44570054 Ki = 24000 nM T74166 CVGP31 44570055 Ki = 6300 nM T74166 CPST94 44570056 Ki = 4900 nM T74166 C0VZ9I 44570057 Ki = 38000 nM T74166 CQ8L9B 44570097 Ki = 100000 nM T74166 CU7S2P 44570098 Ki = 1000000 nM T74166 CFUE82 44570099 Ki = 1000000 nM T74166 C31CSH 44570100 Ki = 100000 nM T74166 CQS02B 44570101 Ki = 39810.72 nM T74166 CMP1K2 44570102 Ki = 39810.72 nM T74166 C2X4GC 44570103 Ki = 31622.78 nM T74166 C18JSV 44570104 Ki = 14000 nM T74166 C7I6OB 44570105 Ki = 12000 nM T74166 C1A2TU 44575473 IC50 > 1000 nM T74166 C5LVN7 44580251 EC50 > 100000 nM T74166 C5Y3MD 44580252 EC50 > 100000 nM T74166 CE85LC 44589967 Ki = 0.2 nM T74166 CVH9T3 44593550 EC50 = 158489.32 nM T74166 C7MB5N 45141377 IC50 = 2 nM T74166 CMSH89 45141378 IC50 = 11 nM T74166 CTL0U6 45141609 IC50 = 15 nM T74166 CQK28Z 45379093 Ki = 390 nM T74166 C6G2TZ 46191426 IC50 > 1000 nM T74166 CQ7S3X 46837648 IC50 = 5600 nM T74166 CL7VN1 46837649 IC50 = 1400 nM T74166 CU7OG4 46837651 IC50 = 11000 nM T74166 C5WNL1 46837652 IC50 = 14000 nM T74166 COX2H5 46837653 IC50 = 20000 nM T74166 CWZY17 46837780 IC50 = 5100 nM T74166 CV2NT3 46837781 IC50 = 8600 nM T74166 CT83MU 46837782 IC50 = 11000 nM T74166 C5TY3Q 46837783 IC50 = 1300 nM T74166 CWJF83 46837784 IC50 = 11900 nM T74166 C0ZSY5 46837785 IC50 = 11000 nM T74166 CBQJ74 46837922 IC50 = 4300 nM T74166 C8UWQ2 46837923 IC50 = 3100 nM T74166 CCX8T0 46837924 IC50 = 2800 nM T74166 CBH49N 46837925 IC50 = 4600 nM T74166 CE71GL 46846404 Ki = 102 nM T74166 C3K6HF 46877888 Ki = 700 nM T74166 C5G7QD 47461992 IC50 = 65500 nM T74166 CXC5S7 49780346 EC50 = 1350 nM T74166 CP8E4O 49788655 IC50 = 2.63 nM T74166 CMI0J4 49788727 IC50 = 2.19 nM T74166 CU8O9W 49788729 IC50 = 2.83 nM T74166 C9QH1W 49788731 IC50 = 0.16 nM T74166 C2UO0F 49799236 IC50 > 100000 nM T74166 C6FH8G 49799237 IC50 > 100000 nM T74166 CZ76MQ 49799633 IC50 = 2600 nM T74166 CU28RO 49799634 IC50 = 3900 nM T74166 CN89XG 49799642 IC50 = 5200 nM T74166 C85MBT 49799643 IC50 = 2000 nM T74166 C5TH3U 49859909 EC50 > 316227.77 nM T74166 CR53VH 49862169 Ki = 1.21 nM T74166 C8WRF4 49862171 Ki = 16.9 nM T74166 C5N4VK 49862173 Ki = 0.882 nM T74166 CX94UB 49862175 EC50 = 32.7 nM T74166 C15OJH 49862213 Ki = 2.1 nM T74166 CT3WH4 49862215 Ki = 0.186 nM T74166 C15JDC 49862217 Ki = 2.02 nM T74166 CC97JM 49862219 Ki = 0.856 nM T74166 CT39UZ 49862259 Ki = 2.17 nM T74166 CTYH68 49862261 Ki = 0.957 nM T74166 CHBT02 49862263 Ki = 1.48 nM T74166 C47WAJ 49862265 Ki = 0.382 nM T74166 CV96ZG 49862267 Ki = 0.158 nM T74166 CQ38SD 49862303 Ki = 1.33 nM T74166 CL7KG5 49862305 Ki = 0.149 nM T74166 C9G7LW 49862307 Ki = 0.126 nM T74166 CGI23Z 49862361 Ki = 9.53 nM T74166 CAI26L 49862363 Ki = 3.79 nM T74166 CO7BM6 49862364 Ki = 496 nM T74166 C2RY0J 50878551 Ki > 10000 nM T74166 CL2P8X 52920232 EC50 > 100000 nM T74166 C42ROG 52920234 EC50 > 100000 nM T74166 CCP0V7 52920236 EC50 > 100000 nM T74166 CU2WT8 52941697 IC50 = 2.62 nM T74166 C3AKS2 53302872 Ki = 2.64 nM T74166 CJ3D7I 53483934 IC50 > 10000 nM T74166 CJ34EQ 53483935 IC50 = 1800 nM T74166 CEY2B8 54583277 IC50 = 790 nM T74166 C6ME0B 54584239 IC50 = 980 nM T74166 CQ71VT 56643499 Ki = 310 nM T74166 C5BJ6G 56648852 Ki = 310 nM T74166 CTS0X9 56649608 Ki = 6600 nM T74166 CLH24J 56663402 IC50 > 10000 nM T74166 CU7OP3 56666825 IC50 > 10000 nM T74166 CY01LS 56666826 IC50 > 10000 nM T74166 CCP40B 56666827 IC50 > 10000 nM T74166 CVT85Q 56670262 IC50 = 1050 nM T74166 C7XK8I 56677105 IC50 = 2900 nM T74166 C02AZR 56677106 IC50 > 10000 nM T74166 C3H1PQ 56835059 IC50 = 23800 nM T74166 CW24DK 56924658 Ki = 4.6 nM T74166 C6V5XD 56926498 IC50 > 100000 nM T74166 C8BOP0 56926617 IC50 > 100000 nM T74166 C94PJS 56926722 IC50 > 100000 nM T74166 C06NVX 56926723 IC50 > 100000 nM T74166 CQ0GH2 56926724 IC50 = 23800 nM T74166 C1TEQ0 56926725 IC50 = 23500 nM T74166 CGP8Q5 56949921 Ki = 7.3 nM T74166 CIC7O5 56950047 Ki = 129 nM T74166 CEG4N8 57334716 EC50 > 100000 nM T74166 CT75BQ 57390841 IC50 = 9400 nM T74166 C20KGJ 57390893 IC50 = 22387.21 nM T74166 C76VTP 57390894 IC50 = 8128.31 nM T74166 C5CG8V 57390895 IC50 = 389045.14 nM T74166 CID85U 57392658 IC50 = 331131.12 nM T74166 CC7R8I 57394370 IC50 = 39600 nM T74166 CLH9Z5 57394409 IC50 = 13803.84 nM T74166 C83BUR 57396127 IC50 = 2700 nM T74166 CK4F0Z 57396175 IC50 = 100000000 nM T74166 CBJ4O8 57397943 IC50 = 10471.29 nM T74166 CO75FJ 57397988 IC50 = 63095.73 nM T74166 CUN0R4 57399583 IC50 = 15488.17 nM T74166 C40FXL 57399584 IC50 = 6300 nM T74166 C2DTL4 57399630 IC50 = 6456.54 nM T74166 CTEP10 57399631 IC50 = 1819.7 nM T74166 CO2MZ8 57399632 IC50 = 4265.8 nM T74166 CU8JW6 57399634 IC50 = 40738.03 nM T74166 C9UMV6 57401339 IC50 = 7244.36 nM T74166 C1WHQ4 57401340 IC50 = 6000 nM T74166 C83MZY 57401393 IC50 = 4786.3 nM T74166 CX4T1A 57403094 IC50 = 10232.93 nM T74166 C9UQF0 57403142 IC50 = 15488.17 nM T74166 C8PHB9 57403143 IC50 = 6606.93 nM T74166 C9K4SR 57403146 IC50 = 14454.4 nM T74166 CV31DZ 57485530 Ki = 12 nM T74166 CZ4G2Y 57485620 Ki = 58 nM T74166 C9G5JE 57485797 Ki = 4.8 nM T74166 CR2V6D 57485798 Ki = 17 nM T74166 CG1TP6 57485799 Ki = 1.9 nM T74166 CON1Z4 57485800 Ki = 14.3 nM T74166 CDW7N1 57486266 Ki = 328 nM T74166 CCM98N 57486336 Ki = 6.2 nM T74166 C50EUG 58006940 Ki = 3800 nM T74166 COT69D 58081856 EC50 > 100000 nM T74166 CE8V0W 58081870 EC50 > 100000 nM T74166 C9V8HI 58088056 EC50 > 100000 nM T74166 CMY5N3 58088118 EC50 > 100000 nM T74166 CP15TC 58201402 Ki = 1200 nM T74166 CW03VZ 58201405 Ki = 380 nM T74166 CP47JL 58201407 Ki = 860 nM T74166 CMKN28 58201409 Ki = 36 nM T74166 CP8G5N 58201418 Ki = 810 nM T74166 C0TML6 58201419 Ki = 150 nM T74166 CB32IW 58201420 Ki = 420 nM T74166 CRC51J 58201424 Ki = 320 nM T74166 C2XCI7 58312740 Ki = 15000 nM T74166 C3KJ7N 58488107 Ki = 420 nM T74166 COQ52A 59268918 Ki = 6600 nM T74166 C4S7VM 59268924 Ki > 10000 nM T74166 CYV48O 59268925 Ki = 12000 nM T74166 C4N2FX 59268932 Ki = 1100 nM T74166 CSW42A 59268935 Ki > 10000 nM T74166 CVN48B 59268936 Ki = 7100 nM T74166 CYSC50 59268939 Ki = 9300 nM T74166 CTR7E8 59268940 Ki = 6500 nM T74166 CHR48L 59268945 Ki = 22000 nM T74166 C1TJ6W 59268948 Ki = 8300 nM T74166 C3EJ6I 59268964 Ki = 7700 nM T74166 CT61RD 59268965 Ki = 3200 nM T74166 C9OS6X 59361675 Ki = 1500 nM T74166 C1J5PV 59361705 Ki = 1700 nM T74166 C6OJH7 59403341 Ki = 2200 nM T74166 CP3XT2 64204965 Ki > 1000 nM T74166 CS67GH 64204975 Ki > 1000 nM T74166 CX90RF 66211794 Ki = 21000 nM T74166 CXN68J 66212381 Ki = 4400 nM T74166 CXR63E 66212976 Ki = 14000 nM T74166 C65UFK 66213161 Ki = 8400 nM T74166 CX9CW1 67585976 Ki = 793 nM T74166 CRSX31 68024489 Ki = 21000 nM T74166 CPA38K 68024616 Ki = 3200 nM T74166 CGU14E 68024620 Ki > 10000 nM T74166 C38FDK 68024820 Ki = 4800 nM T74166 CR0Q4N 68465506 Ki = 70 nM T74166 C1HA9T 68845701 Ki = 155 nM T74166 CF9TX0 69604735 Ki = 21 nM T74166 C5G0FN 69629839 Ki = 6.1 nM T74166 CE0N4K 70675110 Ki = 3.09 nM T74166 C0DX3I 71449982 Ki = 7234 nM T74166 C5BH6L 71450029 Ki = 1831 nM T74166 CQE53F 71450030 Ki = 26 nM T74166 CY5XZ3 71450042 EC50 > 1000 nM T74166 C96JMX 71450130 Ki = 1500 nM T74166 C2I4CF 71450171 Ki = 200 nM T74166 CRX2E6 71451808 Ki = 986 nM T74166 CQ5XI6 71451809 Ki = 507 nM T74166 C9J0NM 71451810 Ki = 4 nM T74166 C5SX4G 71451811 Ki = 1726 nM T74166 CZ42AI 71451812 Ki = 8.3 nM T74166 CB6V1U 71451813 Ki = 40 nM T74166 C9DH7V 71451944 Ki = 14000 nM T74166 CJ01HW 71451994 Ki = 110 nM T74166 CI8YM0 71453627 Ki = 31 nM T74166 C1OS8W 71453628 Ki = 103 nM T74166 C89KME 71453629 Ki = 79 nM T74166 CDGO46 71453630 Ki = 17 nM T74166 C3UW8E 71453631 Ki = 1796 nM T74166 C91CNU 71453666 Ki = 15 nM T74166 C7EU0L 71453717 EC50 > 1000 nM T74166 C3EBR5 71453718 EC50 > 1000 nM T74166 CV0Q4C 71453769 Ki = 8700 nM T74166 CJL26M 71453770 Ki = 3000 nM T74166 CE96BS 71455355 Ki = 56 nM T74166 CLX57K 71455356 Ki = 534 nM T74166 CNGK53 71455357 Ki = 596 nM T74166 C8N4IJ 71455358 Ki = 711 nM T74166 CDC54A 71455359 Ki = 1639 nM T74166 CQMZ91 71455409 IC50 > 1000 nM T74166 C4SRA8 71455410 EC50 > 1000 nM T74166 CYJT51 71455446 IC50 > 1000 nM T74166 C5MFX7 71455447 EC50 > 1000 nM T74166 C8Z4ES 71455499 Ki = 27000 nM T74166 CFOH06 71455500 Ki = 5200 nM T74166 CT79WZ 71455501 Ki = 900 nM T74166 C71PCM 71455535 Ki = 450 nM T74166 CFMS41 71457131 Ki = 459 nM T74166 CO5B7Z 71457133 Ki = 28 nM T74166 CK10DR 71457134 Ki = 23 nM T74166 CCFH76 71457135 Ki = 8.2 nM T74166 CY4U7W 71457136 Ki = 39 nM T74166 CYA78X 71457185 EC50 > 1000 nM T74166 C0Y4UB 71457186 EC50 > 1000 nM T74166 CH84SU 71457187 EC50 > 1000 nM T74166 CS8Q5A 71457513 Ki = 6100 nM T74166 CN0AH1 71458995 Ki = 73 nM T74166 C7V0CY 71458996 EC50 = 1890 nM T74166 CH7U6N 71458997 Ki = 44 nM T74166 CUC0T8 71458998 Ki = 5.4 nM T74166 C96NIY 71459035 Ki = 15 nM T74166 C1WME8 71459126 Ki = 600 nM T74166 CU5D0T 71460792 Ki = 1305 nM T74166 CW58SI 71460793 Ki = 25 nM T74166 CU7CZ6 71460794 Ki = 4502 nM T74166 CZKD91 71460795 Ki = 1431 nM T74166 CWJ1I2 71460832 Ki = 47 nM T74166 C0G4SZ 71460833 Ki = 22 nM T74166 C5TSZ4 71460834 Ki = 27 nM T74166 C2C1JW 71460847 EC50 > 1000 nM T74166 CUXK17 71460848 EC50 > 1000 nM T74166 CKM9O5 71460849 EC50 > 1000 nM T74166 CWE61H 71460892 EC50 > 1000 nM T74166 CV37ZJ 71462520 Ki = 40 nM T74166 C86IYC 71462521 Ki = 5736 nM T74166 CFD1B9 71462522 Ki = 828 nM T74166 C3YZ6W 71462523 Ki = 128 nM T74166 CK3N6Z 71462524 Ki = 7 nM T74166 CX6V7B 71462553 EC50 > 1000 nM T74166 CUP15I 71462588 EC50 > 1000 nM T74166 CM0HG2 71462689 Ki = 1700 nM T74166 CJ7ER8 71682669 Ki = 2000 nM T74166 C05CTI 71682670 Ki = 280 nM T74166 CMKP08 71682671 Ki = 360 nM T74166 CT34ZA 71682672 Ki = 13000 nM T74166 C5BO6T 71682826 EC50 = 1300 nM T74166 CAG7D4 71682974 EC50 = 100000 nM T74166 C9C3EG 71682975 Ki = 4000 nM T74166 C20NXV 71682976 Ki = 6000 nM T74166 C3DXJ1 71718802 IC50 = 602.56 nM T74166 CRU4E7 71720631 Ki = 2100 nM T74166 C7W1RU 71727769 IC50 > 100000 nM T74166 CQJ70U 71727770 IC50 = 27400 nM T74166 C35IOD 71727771 IC50 > 100000 nM T74166 CCF6M0 71727772 IC50 > 100000 nM T74166 CMT9S5 71727773 IC50 = 22500 nM T74166 CI01GP 71727774 IC50 = 29200 nM T74166 C52MJY 71727775 IC50 = 12600 nM T74166 C3NK1F 71727895 IC50 = 77800 nM T74166 CW72HR 71727896 IC50 > 100000 nM T74166 C7INR8 71727897 IC50 > 100000 nM T74166 CJZ5K9 71727898 IC50 > 100000 nM T74166 CJYM35 71727899 IC50 > 100000 nM T74166 CQ24PX 71727900 IC50 > 100000 nM T74166 C08YLD 71727901 IC50 > 100000 nM T74166 C17IXA 71728020 IC50 > 100000 nM T74166 C6F3NV 71728021 IC50 > 100000 nM T74166 C3FZ8C 71728022 IC50 > 100000 nM T74166 C8OGQ1 71728023 IC50 > 100000 nM T74166 CE1Z0Y 71728024 IC50 = 11700 nM T74166 CO4G6R 71728025 IC50 = 19200 nM T74166 CHW18L 72703052 Ki = 9000 nM T74166 C6NOM3 72703256 Ki = 709 nM T74166 C0GQ7F 72703471 Ki = 5000 nM T74166 CMZ19D 72703472 Ki = 3000 nM T74166 CCE9W7 72703473 Ki = 261 nM T74166 CY56RE 73347561 Ki = 100 nM T74166 C71LER 73350667 Ki = 10 nM T74166 CER79N 73352166 Ki = 600 nM T74166 CIX69R 73353186 IC50 = 5 nM T74166 CYL5C0 73355120 Ki = 100 nM T74166 CKD42Z 75113427 Ki = 11 nM T74166 C3CH5U 76310142 IC50 = 97 nM T74166 CF5OB2 76324742 IC50 = 3390 nM T74166 CU89CH 76328290 IC50 = 755 nM T74166 CXT06Q 77139555 Ki > 1000 nM T74166 CPHO43 77907039 Ki = 8.5 nM T74166 CZCV56 89943572 Ki = 1010 nM T74166 CUX53L 89943718 Ki = 362 nM T74166 CEI2S7 89943719 Ki = 5.24 nM T74166 CHYU63 90654473 IC50 = 2.3 nM T74166 CI0W1V 90654475 IC50 = 97 nM T74166 C91DCW 90654485 IC50 = 755 nM T74166 C0UYS5 122182084 Ki > 1000 nM T74166 CQ90NE 122182085 Ki > 1000 nM T74166 C14TQD 122182202 Ki > 1000 nM T74166 C8FZM1 122182203 Ki > 1000 nM T74166 CK1EV8 122182204 Ki > 1000 nM T74166 COAE62 122182205 Ki > 1000 nM T74166 C3Q7RB 122182206 Ki > 1000 nM T74166 CIM90P 122182207 Ki > 1000 nM T74166 CO5G3C 122182208 Ki > 1000 nM T74166 CT8EG2 122182209 Ki > 1000 nM T74166 CK9CR6 122182210 Ki > 1000 nM T74166 C0FRG8 122182211 Ki > 1000 nM T74166 CZ4A6T 122182213 Ki > 1000 nM T74166 C6FY0M 122182214 Ki > 1000 nM T74166 C8GC5V 122182215 Ki > 1000 nM T74166 CF5H7Z 122182216 Ki > 1000 nM T74166 C01YCG 122182217 Ki > 1000 nM T74166 C2TO8V 122185335 Ki = 74 nM T74166 CKCS30 122185336 Ki = 102 nM T74166 C3TWG2 122185337 Ki = 40 nM T74166 CDQO08 122185338 Ki = 235 nM T74166 CTS5K0 122185339 Ki = 100 nM T74166 CZHP50 122185340 Ki = 1300 nM T74166 CAR46I 122185341 Ki = 1400 nM T74166 CR3E5H 122185342 Ki = 271 nM T74166 C7C4EN 122185343 Ki = 7700 nM T74166 C6QDM0 122185344 Ki = 257 nM T74166 CD3ET9 122185345 Ki = 752 nM T74166 CKOG84 122185346 Ki = 5300 nM T74166 C1LID2 122185347 Ki = 2100 nM T74166 CZ2IM4 122185348 Ki = 2900 nM T74166 CXVF35 122185349 Ki = 5000 nM T74166 CUAI92 122185350 Ki = 5600 nM T74166 C6LHN9 122193497 Ki = 2.6 nM T74166 CTC87H 122193500 Ki = 1.6 nM T74166 CR0P7N 122553341 Ki = 3.44 nM T74166 C19IZT 127024854 Ki = 29.8 nM T74166 CKMX40 127026063 Ki = 80 nM T74166 CHIT14 127026744 Ki = 77.2 nM T74166 C39VRU 127026745 Ki = 70.8 nM T74166 C9QBZ8 127026746 Ki = 48 nM T74166 C2RQ0I 127027053 Ki = 80 nM T74166 CC7X3R 127027054 Ki = 92 nM T74166 CVOQ45 127027055 Ki = 80 nM T74166 C4XDC6 127028296 Ki = 4.7 nM T74166 C4FT9P 127028304 Ki = 680 nM T74166 CHB8E5 134137043 Ki = 415 nM T74166 CE0Z1P 134138340 Ki = 122 nM T74166 CX9A0R 134139125 Ki = 947 nM T74166 CK31WO 134139695 Ki = 1200 nM T74166 CMVN28 134140850 Ki = 200 nM T74166 C8AX7R 134141073 Ki = 3100 nM T74166 CK7SL8 134142202 Ki = 8300 nM T74166 CVYC45 134144007 Ki = 147 nM T74166 C8MQ6C 134157065 Ki = 30 nM T74166 CLE38V 135508231 Ki = 970 nM T74166 CX0LF6 137633214 EC50 > 100000 nM T74166 C93ZPK 137635141 EC50 > 100000 nM T74166 CTU9Y7 137635902 EC50 > 100000 nM T74166 C3QA9I 137637512 Ki = 5800 nM T74166 C3UT9L 137643408 EC50 > 100000 nM T74166 CVJ0Q7 137644763 EC50 > 100000 nM T74166 C9K7VP 137644928 EC50 > 100000 nM T74166 CPCY48 137645406 Ki = 8523 nM T74166 CQ5H2Y 137645815 EC50 > 100000 nM T74166 CV9T6B 137647317 EC50 > 100000 nM T74166 C3Y2SW 137649484 EC50 > 100000 nM T74166 CA8L7Z 137649750 Ki = 8900 nM T74166 C6RJ8V 137649905 EC50 > 100000 nM T74166 C5U0GB 137650643 Ki = 22000 nM T74166 CCY0D8 137652873 Ki = 16200 nM T74166 CVON14 137654242 EC50 > 100000 nM T74166 CJC95L 137654434 EC50 > 100000 nM T74166 COVD20 137655697 EC50 > 100000 nM T74166 C6CYW8 137657023 EC50 > 100000 nM T74166 CS3K4D 137659736 EC50 > 100000 nM T74166 CX39HQ 137659815 EC50 > 100000 nM T74166 C4GOE0 137660090 EC50 > 100000 nM T74166 CP48RG 137660174 EC50 > 100000 nM T74166 C0B6HQ 137660214 EC50 > 100000 nM T74166 C3FZL5 141725921 IC50 = 10080 nM T74166 CM5EY7 145949363 Ki = 1.2 nM T74166 C4Q8CK 145949640 Ki = 165 nM T74166 CIPU07 145949810 Ki = 40.9 nM T74166 CN8KT3 145951677 Ki = 0.988 nM T74166 CG39CO 145954266 Ki = 1.25 nM T74166 C43URC 145954515 Ki = 25 nM T74166 CB5XT1 145955237 Ki = 115 nM T74166 C69IDF 145955461 Ki = 1.02 nM T74166 C2CSF8 145955621 Ki = 0.799 nM T74166 CH8KS9 145957714 Ki = 293 nM T74166 C69FXT 145958303 Ki = 1.4 nM T74166 C4U1CR 145959650 Ki = 4.8 nM T74166 CZ48DQ 145960008 Ki = 0.818 nM T74166 C6UZJ9 145960066 Ki = 9.03 nM T74166 CDI60M 145960262 Ki = 0.684 nM T74166 CCX4T1 145964547 Ki = 123 nM T74166 CAP3V1 145971759 Ki = 13 nM T74166 COY76F 145972407 Ki = 2.2 nM T74166 C7XB0C 145989786 Ki = 9.1 nM T74166 C6Q3XK 146680925 Ki = 1090 nM T74166 C6DCN9 146680926 Ki = 2.25 nM T74166 CAE65X 155510505 Ki = 21 nM T74166 CDA38T 155511206 Ki = 103 nM T74166 C9F6LV 155512339 Ki = 20.9 nM T74166 CM7DV8 155514108 IC50 = 0.95 nM T74166 CT64LK 155514460 Ki = 19.5 nM T74166 C5AS9Y 155515572 Ki = 59 nM T74166 CMV2G7 155515603 Ki = 7.17 nM T74166 C7DBH6 155516230 Ki = 11.8 nM T74166 CW8IV5 155516492 IC50 = 0.55 nM T74166 C7PHA3 155517726 Ki = 113 nM T74166 C7P0NK 155518882 Ki = 123 nM T74166 C5GAS9 155521191 Ki = 6.67 nM T74166 CHC38D 155522533 Ki = 44.4 nM T74166 CK01QX 155522758 Ki = 2.48 nM T74166 CE8UV4 155522802 Ki = 102 nM T74166 C19POZ 155523848 IC50 = 0.37 nM T74166 C5U6IO 155527752 Ki = 81 nM T74166 CFAY97 155528499 IC50 = 960 nM T74166 C2YXJ9 155529181 IC50 = 0.35 nM T74166 C4JPE6 155529322 Ki = 516 nM T74166 C57HKR 155529699 IC50 = 0.65 nM T74166 CLYV89 155530137 Ki = 631 nM T74166 C3VOB7 155532967 Ki = 1628 nM T74166 CO07HD 155533348 Ki = 7.57 nM T74166 CIGK42 155536100 Ki = 1600 nM T74166 CMK0U4 155537399 Ki = 558 nM T74166 CH38YT 155538341 Ki = 306 nM T74166 C8Y4PI 155541561 IC50 = 1.44 nM T74166 CI54SN 155544676 Ki = 28 nM T74166 CL8I6H 155545841 Ki = 2000 nM T74166 CD3EW6 155546334 IC50 = 0.92 nM T74166 C7W5ZC 155547147 Ki = 265 nM T74166 CM50TS 155547626 Ki = 138 nM T74166 CROV92 155554398 Ki = 13.9 nM T74166 CX2U1M 155556961 Ki = 50 nM T74166 C6RU4P 155557819 IC50 = 1.07 nM T74166 CQ52KG 155561319 Ki = 62 nM T74166 C9HAJ3 155562518 Ki = 192 nM T74166 CW51RT 155564442 IC50 = 0.57 nM T74166 CB0LH8 11602721 IC50 = 1000 nM T74166 CTAK49 11660066 IC50 = 794.33 nM T74166 C7NWZ6 442202 IC50 = 1780 nM T74166 CUZ1D8 44564663 IC50 = 1000 nM T74166 D00GDI 45487890 IC50 = 6.8 nM T74166 D00QCP 46837647 IC50 = 8900 nM T74166 D01YED 45141808 IC50 = 16 nM T74166 D02ZIQ 43227131 IC50 = 7.7 nM T74166 D03YQY 46837650 IC50 = 8600 nM T74166 D04KZX 44542809 IC50 = 0.51 nM T74166 D05PLF 3031066 IC50 = 2.4 nM T74166 D06LCK 45141805 IC50 = 35 nM T74166 D08SCF 159548 IC50 = 7.65 nM T74166 D09BYB 45487941 IC50 = 2.4 nM T74166 D09XWL 45141379 IC50 = 11 nM T74166 D0C0GL 3031062 IC50 = 1.3 nM T74166 D0G0CJ 45141380 IC50 = 3.9 nM T74166 D0G1XP 44543273 IC50 = 0.62 nM T74166 D0GY8R 45141807 IC50 = 11 nM T74166 D0H4AD 44542509 IC50 = 1.4 nM T74166 D0IP9V 10107234 IC50 > 100000 nM T74166 D0J5EF 215051 IC50 = 4.4 nM T74166 D0O2LC 44543272 IC50 = 26 nM T74166 D0O5EZ 854023 Ki = 0.15 nM T74166 D0P9EO 45141381 IC50 = 3.7 nM T74166 D0Q8IQ 43794735 IC50 = 37 nM T74166 D0R4RN 1204 Ki = 0.15 nM T74166 D0R8EV 3027752 IC50 = 0.58 nM T74166 D0U3SB 45141806 IC50 = 11 nM T74166 D0V0AW 9823180 Ki = 7000 nM T74166 D0VY9K 45141809 IC50 = 53 nM T74166 D0X7HD 11184481 Ki = 5370 nM T74166 D0XY9E 3029724 IC50 = 0.7 nM T74166 D0Y7CS 44543118 IC50 = 1.5 nM T74166 D0ZE4C 45141608 IC50 = 4.7 nM T00973 C2M0SE 1511198 IC50 > 100000 nM T00973 CJK1F0 1511199 IC50 > 100000 nM T00973 CR3SF5 4907545 IC50 > 100000 nM T00973 CWG19Q 4908238 IC50 > 100000 nM T00973 CG3PR6 52912222 IC50 = 630.96 nM T00973 CIPN50 71760902 IC50 > 1000 nM T00973 C5TB9S 77843982 IC50 > 10000 nM T00973 COZ8S1 78319129 IC50 > 1000 nM T00973 CUWX94 119081692 IC50 = 7600 nM T00973 CVBC47 155535120 Ki = 2500 nM T83813 D00JVR 2267 Ki = 501.19 nM T83813 D00TLN 2913 Ki = 11 nM T83813 D00XWD 135409453 Ki < 100 nM T83813 D01AZG 5073 IC50 = 1.81 nM T83813 D01JMC 11658860 EC50 = 1.82 nM T83813 D01ZII 2726 Ki = 27 nM T83813 D03WEX 9966051 Ki = 180 nM T83813 D04JEE 4946 EC50 > 5011.87 nM T83813 D05ZIK 4205 Ki = 39 nM T83813 D06XZR 27400 Ki = 1.4 nM T83813 D06ZUK 3696 Ki = 160 nM T83813 D08VRO 3822 IC50 = 2.7 nM T83813 D0CQ0Z 33630 Ki = 881 nM T83813 D0D1AL 3559 Ki = 2511.89 nM T83813 D0F2PO 4828 Ki = 54000 nM T83813 D0H3HM 60795 Ki = 22 nM T83813 D0H7KF 5002 Ki > 1000 nM T83813 D0O6GC 9681 Ki = 2.5 nM T83813 D0R1JV 60854 Ki = 0.55 nM T83813 D0R6RO 4184 Ki = 1.7 nM T83813 D0S9MU 5078 IC50 = 7943.28 nM T83813 D0T6QX 5736 Ki = 2.9 nM T83813 D0U2OO 2477 Ki = 2270 nM T83813 D0UA0I 28693 Ki = 0.5 nM T83813 D0V4QS 135398745 Ki = 2.8 nM T83813 D0W5HK 216239 Ki = 417 nM T83813 D0YG7M 3827 Ki = 199.53 nM T83813 D0Z1RV 135398737 Ki = 2.884 nM T83813 D0Z6UC 5358 IC50 = 7.3 nM T83813 D00TLM 6433122 Ki = 645 nM T83813 D02BRJ 11521822 Ki = 3 nM T83813 D04GMY 11842633 Ki < 100 nM T83813 D08CJK 1150 Ki = 50 nM T83813 D09IRN 21071390 Ki = 250 nM T83813 D0GJ7B 11683556 Ki = 110 nM T83813 D0HZ2E 5311271 Ki = 13 nM T83813 D0LI1C 44469321 IC50 > 10000 nM T83813 D0N1HW 5311200 Ki > 10000 nM T83813 D0R9KG 11604525 Ki > 10000 nM T83813 D0U0KR 3035850 Ki = 10000 nM T83813 D0Y6ZK 123683 Ki = 5420 nM T83813 D00OWF 5280953 Ki = 9340 nM T83813 D00PXQ 60785 Ki = 1 nM T83813 D02JMI 9888211 Ki = 39.81 nM T83813 D02ZSO 6426760 IC50 = 9000 nM T83813 D03PJW 108029 IC50 = 290 nM T83813 D03YPJ 5163 IC50 = 9.4 nM T83813 D04DGE 9888804 Ki = 0.5012 nM T83813 D05MFO 71781 Ki = 10000 nM T83813 D06DZI 107780 Ki = 105 nM T83813 D06ZVC 10150497 Ki = 124 nM T83813 D08AWI 11430856 Ki > 5000 nM T83813 D0B4BN 3045227 Ki = 1.259 nM T83813 D0B7SP 11292933 Ki = 1584.89 nM T83813 D0G1RT 132059 IC50 = 316.23 nM T83813 D0K8NW 5074 Ki = 0.71 nM T83813 D0K9JP 9928332 Ki > 1000 nM T83813 D0M7LV 5761 Ki = 5.012 nM T83813 D0OS6O 60149 Ki = 0.2 nM T83813 D0Q2JS 10436045 Ki = 79.43 nM T83813 D0S5FQ 7153 EC50 = 120 nM T83813 D0U7VZ 11225102 Ki < 100 nM T83813 D0Y8UB 82148 Ki = 630 nM T83813 D0YP7L 6604889 Ki < 5 nM T83813 C5JG6U 2689 IC50 > 10000 nM T83813 C5H9CN 9287 EC50 = 107.1 nM T83813 C6KIN7 10624 EC50 = 506 nM T83813 CW3P5L 11297 Ki = 40 nM T83813 CHF8L6 12834 Ki = 10 nM T83813 C7VE9O 27557 Ki = 6.1 nM T83813 CR69PX 29101 Ki = 540 nM T83813 C4RF5C 30241 Ki = 1 nM T83813 CF3R1X 38240 Ki = 177.2 nM T83813 C6KXM1 62857 Ki = 72 nM T83813 CG02IV 82509 Ki > 10000 nM T83813 CB6G3Z 91536 Ki = 1400 nM T83813 CKP25M 121881 Ki = 79.43 nM T83813 C4PR2E 132564 IC50 = 100 nM T83813 CFV6Z2 150885 Ki = 280 nM T83813 C93TIV 160463 Ki = 5500 nM T83813 CGT8R0 160510 Ki = 1860 nM T83813 CLK7P3 169713 IC50 = 1290 nM T83813 CF5WT9 171289 Ki > 300000 nM T83813 CX7SJ2 334449 IC50 = 1050 nM T83813 C68WUF 395901 Ki > 10000 nM T83813 CYV1R3 417052 Ki = 924 nM T83813 CJ6X4W 498210 Ki = 23 nM T83813 C24IFT 544738 Ki = 1800 nM T83813 C4KIJ8 544751 Ki > 10000 nM T83813 CMT84S 603606 EC50 = 9 nM T83813 CPI69B 702235 EC50 = 128 nM T83813 CQW20U 715057 IC50 = 2534 nM T83813 CMIS59 715058 IC50 = 1863 nM T83813 CXQ6U0 735755 IC50 = 2500 nM T83813 CZN6S9 743974 EC50 > 39810.72 nM T83813 C2VLP8 752521 Ki = 265 nM T83813 CU0H9A 1129292 IC50 = 1208 nM T83813 C6EYN9 1203613 Ki > 10000 nM T83813 CYE02G 1400243 EC50 = 3162.28 nM T83813 CVXJ06 1497577 EC50 = 16 nM T83813 C0TQ8H 2407992 IC50 = 1055 nM T83813 C46RBT 2444416 IC50 = 179 nM T83813 C1MD9K 2723612 EC50 = 1760 nM T83813 C3RWU0 2723860 EC50 = 2450 nM T83813 CO5U6X 2759136 Ki > 10000 nM T83813 CPI2C5 2775690 Ki = 965 nM T83813 C9IBF5 2955320 IC50 > 10000 nM T83813 C2RZW5 2976205 IC50 > 10000 nM T83813 CJ14KW 2997467 IC50 > 10000 nM T83813 C64CZV 3038494 Ki = 218 nM T83813 C2F7ZC 3045234 Ki = 2.512 nM T83813 C4R0OH 3045236 Ki = 2.512 nM T83813 C1FV0B 3045239 Ki = 1 nM T83813 CAM8H3 3066250 IC50 > 1000 nM T83813 CS5F1I 3083481 Ki = 230 nM T83813 CNX8I1 3245407 IC50 = 2900 nM T83813 C69OAZ 3434273 IC50 > 10000 nM T83813 CS8KE2 3649661 Ki = 851 nM T83813 C0YXV3 3676358 Ki > 10000 nM T83813 CO75SE 3731509 IC50 = 471 nM T83813 C56JID 3763575 Ki = 8 nM T83813 CN5YK3 3852202 IC50 = 99 nM T83813 CTH61F 3868902 IC50 > 10000 nM T83813 CXD2W7 3870140 IC50 = 766 nM T83813 CK36GS 3906894 Ki = 4 nM T83813 CY67TC 5281073 Ki = 0.7943 nM T83813 CD7U8Z 5311422 Ki = 109.65 nM T83813 C4DCR0 5745501 Ki = 1 nM T83813 CAO47E 6452095 Ki = 9.3 nM T83813 CJL3P7 6473290 IC50 > 10000 nM T83813 C3A1FO 6604789 Ki = 15848.93 nM T83813 C91WQS 6604916 Ki = 3 nM T83813 C7H9MB 6604933 EC50 = 261 nM T83813 CT82ZY 6625601 IC50 > 10000 nM T83813 C0QCK1 6918455 Ki = 1995.26 nM T83813 C1WXY3 6918603 Ki < 2511.89 nM T83813 CD0Z4I 6918648 Ki = 501.19 nM T83813 C8AL9V 6918689 Ki < 10000 nM T83813 CBLE17 7208185 IC50 = 1999 nM T83813 CA2U1M 7208267 IC50 = 2732 nM T83813 CFW9V1 7216312 IC50 = 2588 nM T83813 CRWA82 8545974 IC50 = 991 nM T83813 CU3W4K 9044803 IC50 = 213796.21 nM T83813 CC47WV 9794092 Ki = 4.8 nM T83813 CXI18K 9794638 EC50 = 5.7 nM T83813 COHS59 9795468 Ki = 20 nM T83813 CTYZ64 9798764 Ki = 1200 nM T83813 CB5A6I 9799300 Ki = 50.12 nM T83813 CE0DI5 9804612 Ki < 10000 nM T83813 C8XGV3 9804849 IC50 = 900 nM T83813 CNX4F0 9805456 Ki < 3981.07 nM T83813 CZ2WA1 9813163 Ki = 97 nM T83813 CV6LU0 9813187 Ki = 38 nM T83813 CS3HR6 9813866 Ki = 358 nM T83813 CS1K8O 9814315 Ki = 54 nM T83813 CAEQ74 9817866 Ki = 8 nM T83813 C1ZM6Q 9821397 IC50 = 4000 nM T83813 CL38GM 9826580 Ki = 52.7 nM T83813 C0AU9L 9826801 Ki = 60 nM T83813 C38DHN 9834518 Ki = 74 nM T83813 C0H6DZ 9837204 Ki = 131 nM T83813 CQY5S4 9838040 EC50 = 4 nM T83813 CV2A3K 9838959 Ki = 260 nM T83813 CBN06W 9839050 Ki = 0.93 nM T83813 C28HIY 9839057 Ki = 0.02 nM T83813 CWTA61 9839081 Ki = 1 nM T83813 CQAI06 9839494 Ki = 9 nM T83813 C7H8CZ 9839920 Ki = 25.12 nM T83813 C6I4QG 9841032 IC50 = 1737.8 nM T83813 CDOC72 9844378 EC50 = 22 nM T83813 CC24WR 9845261 IC50 > 100000 nM T83813 CNB65K 9848303 Ki = 110 nM T83813 CWJ75T 9849983 Ki = 5.5 nM T83813 CM13ZV 9856041 Ki = 5.5 nM T83813 C0Q6RX 9856443 Ki = 136 nM T83813 CKQ5O7 9856509 Ki = 2.4 nM T83813 C9B2QD 9859144 Ki = 31 nM T83813 C0ZR3E 9861687 IC50 = 5623.41 nM T83813 C0Q6AD 9863611 Ki = 50.12 nM T83813 CI30XR 9865463 Ki = 128 nM T83813 C5WYN4 9865858 Ki = 58 nM T83813 C0W3JF 9866423 Ki = 1.585 nM T83813 C7FBK5 9866660 Ki = 27.54 nM T83813 C19KGY 9869628 Ki = 0.631 nM T83813 C7AB8O 9870053 Ki = 1258.93 nM T83813 CQ4LC2 9872676 Ki = 964 nM T83813 C86NSR 9877758 Ki = 85 nM T83813 C2ZX0B 9877925 Ki = 985 nM T83813 C2ELZ9 9881053 IC50 = 3400 nM T83813 CKS8Z9 9881119 EC50 = 28 nM T83813 CE46QD 9881885 EC50 = 5 nM T83813 C75IFN 9882045 Ki = 91 nM T83813 CF59KP 9882393 Ki = 6.3 nM T83813 C10MKO 9882537 Ki = 160 nM T83813 CZ8C7G 9885279 Ki = 130 nM T83813 C64EOU 9885465 Ki = 25 nM T83813 CIL0R2 9886130 Ki = 223.87 nM T83813 CJW1P5 9888494 Ki = 3311.31 nM T83813 CM52WU 9890119 Ki < 2511.89 nM T83813 CEG1K5 9891002 Ki = 1258.93 nM T83813 C7QMK5 9891617 Ki = 2511.89 nM T83813 CEL29O 9891618 Ki < 5011.87 nM T83813 C6WY0D 9891901 Ki = 411 nM T83813 C3J8GU 9892409 Ki < 3162.28 nM T83813 C7EZ8Q 9899243 Ki = 12 nM T83813 C2P3GS 9899500 Ki = 1.9 nM T83813 CF6OE1 9899545 Ki = 599 nM T83813 CN6E8D 9899546 Ki = 452 nM T83813 C9J6KN 9901423 Ki < 100 nM T83813 C5TA6D 9903398 Ki = 180 nM T83813 CHFP46 9903970 Ki = 2.455 nM T83813 CN3JG8 9904139 Ki = 66.07 nM T83813 CFI97S 9904205 IC50 = 12.3 nM T83813 CUN81Q 9905249 Ki > 10000 nM T83813 CYWQ50 9906447 Ki > 10000 nM T83813 C7JFZ5 9906978 Ki = 1252 nM T83813 C2Z9BL 9908431 Ki = 640 nM T83813 CYZ5N4 9909089 Ki = 3981.07 nM T83813 CTZ48N 9910346 IC50 = 0.53 nM T83813 C3BR6W 9910451 Ki > 4200 nM T83813 C9B3EA 9911844 Ki < 1000 nM T83813 C78MDV 9913554 Ki = 398.11 nM T83813 C1D4BM 9920585 Ki = 721 nM T83813 CS61ZI 9920667 Ki = 13 nM T83813 C6BTZ9 9920815 Ki = 1.7 nM T83813 C4BZ3W 9921116 Ki = 189 nM T83813 CU7JO2 9921840 Ki = 79 nM T83813 CQ3YN1 9927016 IC50 = 3981.07 nM T83813 CVZ18D 9930475 Ki = 501.19 nM T83813 CO6MD4 9931534 Ki = 1 nM T83813 CAQ52T 9932698 Ki = 22 nM T83813 CIP6V7 9932896 IC50 > 1000 nM T83813 CYVZ47 9934284 Ki = 1258.93 nM T83813 CWO45F 9935387 Ki = 630.96 nM T83813 CLYE56 9942836 Ki = 38 nM T83813 CYH3R7 9947817 Ki = 310 nM T83813 C8T1HO 9948670 Ki = 16 nM T83813 C1H4IP 9951008 Ki = 165.96 nM T83813 CKID85 9951964 Ki = 831.76 nM T83813 C4YH2I 9953216 Ki = 280 nM T83813 CKF9X1 9953268 Ki = 100 nM T83813 CK8NR2 9954121 Ki < 1995.26 nM T83813 CHOJ30 9956365 Ki < 1000 nM T83813 CFR41N 9957068 Ki < 7943.28 nM T83813 C3ZL9T 9964963 Ki = 243 nM T83813 CCZP34 9976750 IC50 = 1584.89 nM T83813 C8P1TR 9978065 Ki = 35.48 nM T83813 CFN50J 9978683 Ki > 5000 nM T83813 CC5K4N 9979654 Ki = 3311.31 nM T83813 C76JBU 9981505 Ki = 5.012 nM T83813 CI1F8K 9981671 IC50 = 600 nM T83813 C2USG0 9983031 Ki = 2.512 nM T83813 CL9UJ7 9990808 EC50 = 6.31 nM T83813 C9FBE5 9991444 EC50 = 3.981 nM T83813 C7P2BT 9994008 EC50 = 11 nM T83813 CF0R6B 9995045 IC50 = 251.19 nM T83813 C0J1CD 9998826 Ki = 1260 nM T83813 CJ89IZ 10000788 Ki = 223.87 nM T83813 CYG36Z 10003368 Ki = 6.31 nM T83813 CT2CS3 10003477 Ki = 15.85 nM T83813 CQL12P 10004545 Ki = 1120 nM T83813 C3C0YF 10008294 Ki = 19.95 nM T83813 CLE61D 10015414 EC50 = 4 nM T83813 CE3FH2 10015954 Ki = 346.74 nM T83813 C45HCE 10017554 Ki = 0.3 nM T83813 CEY30Z 10017556 EC50 = 68 nM T83813 C3B4HS 10017993 EC50 = 19 nM T83813 CV7R9F 10020040 Ki > 10000 nM T83813 CK18LT 10020895 Ki = 1900 nM T83813 C8M6IB 10022123 Ki = 416.87 nM T83813 CYT6R9 10022745 Ki = 3630.78 nM T83813 C5X1KG 10022781 Ki = 34.67 nM T83813 C4KIN3 10024430 Ki = 6165.95 nM T83813 C2EUY0 10035109 Ki > 10000 nM T83813 C12LON 10036629 EC50 = 7.943 nM T83813 C2ZO8M 10037962 Ki = 13 nM T83813 C57TZR 10042333 Ki = 503 nM T83813 C2C1XS 10042602 Ki = 14.45 nM T83813 C20EOP 10044334 Ki = 234.42 nM T83813 CUH63M 10046389 Ki = 650 nM T83813 C25WVJ 10047566 IC50 > 1000 nM T83813 C6M1TH 10050022 Ki = 10 nM T83813 CDSQ03 10058473 Ki = 102 nM T83813 CP9A6Q 10061694 IC50 > 10000 nM T83813 CDKW35 10061837 Ki = 89.13 nM T83813 CDA93R 10062435 IC50 = 5011.87 nM T83813 CFM51X 10063283 IC50 = 2511.89 nM T83813 C5PG9D 10064386 EC50 = 2 nM T83813 C4PCO3 10065083 Ki = 4132 nM T83813 C8Z6MA 10067306 IC50 = 477 nM T83813 CC5LY7 10069784 Ki = 588.84 nM T83813 C2JFB1 10072280 Ki = 609 nM T83813 C7IXA4 10072800 Ki = 87.1 nM T83813 CD2RM6 10085260 Ki = 5.96 nM T83813 CQVJ58 10088453 Ki = 44.67 nM T83813 CVK93I 10090424 Ki = 338.84 nM T83813 C63FME 10090486 Ki = 338.84 nM T83813 C8NQ3I 10092649 Ki = 85 nM T83813 CQ24PH 10093238 Ki = 1258.93 nM T83813 CC5IZ2 10103618 Ki = 44.1 nM T83813 C8F9SD 10105208 EC50 = 6.31 nM T83813 C7EMN2 10105553 Ki = 330 nM T83813 C54EYD 10108561 IC50 = 12.59 nM T83813 CKU06X 10108730 IC50 > 10000 nM T83813 CJ1K5Y 10127939 Ki = 1.995 nM T83813 CZ2S7U 10127968 Ki = 7.943 nM T83813 C8ZJ9G 10131066 Ki = 2.7 nM T83813 CJF76C 10150393 Ki = 3.981 nM T83813 CI2X3Y 10151289 Ki = 25.12 nM T83813 C6FEY0 10151426 Ki = 300 nM T83813 C9TQ1J 10159452 IC50 = 36 nM T83813 CP6Q1W 10173403 Ki = 19.95 nM T83813 CN78BA 10176869 Ki = 32 nM T83813 CUJ06B 10194524 Ki = 12.59 nM T83813 CZB8O2 10198481 Ki = 4.3 nM T83813 CED1V2 10199361 Ki = 1000 nM T83813 C46ECI 10216348 Ki = 1090 nM T83813 C02TKP 10216639 Ki = 31.62 nM T83813 CFJY39 10216820 Ki = 50.12 nM T83813 CRNG42 10217207 Ki = 0.7943 nM T83813 C96ARE 10217208 Ki = 10 nM T83813 CV1B7C 10217687 Ki = 39.81 nM T83813 CYAV42 10236153 Ki = 24 nM T83813 CRJ01O 10237852 Ki = 6.31 nM T83813 C6K5ZM 10244251 IC50 = 100 nM T83813 C21CDB 10244831 Ki = 31.62 nM T83813 CVF1E5 10246054 IC50 = 6.166 nM T83813 CSE47M 10247171 IC50 = 3715.35 nM T83813 CG2B7I 10247701 Ki = 64.57 nM T83813 CE79IC 10249506 Ki = 331.13 nM T83813 C4Q2SH 10249573 Ki = 1000 nM T83813 CSPF93 10252272 Ki = 125.89 nM T83813 CKT7U9 10254433 Ki = 10 nM T83813 CD27VE 10255548 Ki = 3.162 nM T83813 CMRA02 10257042 Ki < 3162.28 nM T83813 CC8PX4 10265905 IC50 = 2511.89 nM T83813 CH31DX 10267394 Ki > 10000 nM T83813 COAP98 10287912 Ki = 1.259 nM T83813 C9KDO8 10287924 Ki = 287 nM T83813 CAT4H3 10288601 Ki = 3.162 nM T83813 C3WQ8A 10288693 Ki = 582 nM T83813 CPW71K 10309622 Ki = 1.259 nM T83813 CZVR72 10310067 Ki = 1090 nM T83813 C8XKC0 10310103 Ki > 4200 nM T83813 CU89JD 10314060 Ki > 10000 nM T83813 CA3E4W 10316297 Ki = 54.95 nM T83813 CFWC08 10321945 Ki = 3.162 nM T83813 CRT0J7 10329912 EC50 = 398.11 nM T83813 CE07JM 10330266 Ki = 64 nM T83813 CT4L5Z 10331841 EC50 = 10 nM T83813 CQUG72 10332474 EC50 = 0.23 nM T83813 C84AVJ 10335309 Ki < 6309.57 nM T83813 CJ4B2X 10335310 Ki = 4073.8 nM T83813 C3E5CB 10337773 Ki = 12589.25 nM T83813 CR3J9S 10338282 Ki = 1548.82 nM T83813 CVO3N7 10344176 IC50 = 610 nM T83813 C9IAV3 10346043 Ki > 5011.87 nM T83813 C86INY 10346749 Ki = 6.31 nM T83813 CS24DU 10353268 Ki = 6.3 nM T83813 C4-DEC 10355779 IC50 = 1000 nM T83813 CQLD40 10356829 Ki = 416.87 nM T83813 CZOK29 10367486 Ki = 125.89 nM T83813 CBQ57F 10368126 Ki = 31.62 nM T83813 CC1GT2 10368204 Ki = 15.85 nM T83813 C23KXL 10371119 Ki = 1.585 nM T83813 CUV0T8 10379049 IC50 = 3162.28 nM T83813 CXQJ16 10379099 IC50 = 7943.28 nM T83813 C5LPM8 10379100 IC50 > 10000 nM T83813 CV2G9H 10379910 EC50 = 160 nM T83813 CE1XW6 10380005 IC50 = 1000 nM T83813 CR3KU9 10380133 IC50 > 5000 nM T83813 CDAC63 10381889 IC50 = 1.047 nM T83813 CMZA83 10383646 Ki = 3067 nM T83813 CT78XH 10384138 Ki = 1.995 nM T83813 C69KIB 10385855 IC50 > 10000 nM T83813 CWY94C 10386748 Ki < 10000 nM T83813 CL83KQ 10388797 IC50 = 2000 nM T83813 CESG32 10389978 IC50 = 1600 nM T83813 C1R5GY 10390089 Ki = 1.585 nM T83813 C2T0CR 10400849 IC50 = 3981.07 nM T83813 CA3NO7 10401602 EC50 = 28 nM T83813 CXU73R 10401626 IC50 = 1000 nM T83813 CVQ9E8 10401691 IC50 = 1258.93 nM T83813 C04WGF 10407367 IC50 = 1135 nM T83813 C0ON1Z 10408409 Ki = 1.995 nM T83813 C0HSY3 10409174 Ki = 512.86 nM T83813 CYA49X 10409431 Ki = 19.95 nM T83813 C5PCO9 10410103 Ki = 100 nM T83813 CK6G0O 10413268 Ki = 5.012 nM T83813 C4TPN1 10413595 Ki = 630.96 nM T83813 CYMX90 10414272 Ki = 6.2 nM T83813 CUBX84 10420386 Ki = 9930 nM T83813 C2B0IU 10421236 Ki > 10000 nM T83813 CWD56M 10421850 IC50 = 1258.93 nM T83813 CR4LS0 10430623 Ki > 5000 nM T83813 CS3HX9 10431639 Ki = 380.19 nM T83813 CD7U5I 10433930 Ki = 1000 nM T83813 CNJ4Z9 10435572 Ki = 2.512 nM T83813 CQ1V2Z 10445845 IC50 = 1995.26 nM T83813 CO7IV6 10450593 Ki = 15 nM T83813 C2G0AH 10450758 Ki = 850 nM T83813 C94TVH 10452995 IC50 > 100000 nM T83813 C8TSH1 10454231 Ki = 6.31 nM T83813 CS9R0E 10455878 Ki = 234.42 nM T83813 C07KPU 10456755 IC50 = 1100 nM T83813 CA43RM 10457586 Ki = 12.59 nM T83813 CSV35T 10458193 Ki = 2.512 nM T83813 C2QO7W 10458785 Ki = 3.981 nM T83813 CTED07 10465263 EC50 = 11 nM T83813 C3EH5D 10468253 IC50 = 3162.28 nM T83813 C5LBS7 10472158 IC50 = 44 nM T83813 CRG9T1 10472780 EC50 = 56 nM T83813 CH2O9Q 10473483 Ki = 912.01 nM T83813 C05ZCT 10474964 Ki = 280 nM T83813 C26KCR 10475231 Ki > 1000 nM T83813 CS01JP 10476876 Ki = 3.981 nM T83813 CX13YD 10477339 Ki = 10 nM T83813 CEF2O6 10478367 Ki = 1937 nM T83813 C12RUZ 10479309 Ki = 19.95 nM T83813 CH64LD 10479409 Ki = 5.012 nM T83813 C04TSD 10487869 Ki = 6.31 nM T83813 CGD21U 10491097 Ki = 158.49 nM T83813 CB52TQ 10495305 Ki = 132 nM T83813 C0CH4G 10495578 Ki = 19.95 nM T83813 CPG8U3 10495787 Ki = 50 nM T83813 C0QR2H 10496957 IC50 > 100000 nM T83813 CKPH17 10497359 Ki < 10000 nM T83813 C38ZFO 10498110 Ki = 6.31 nM T83813 C3IY9P 10498554 IC50 = 57543.99 nM T83813 C4XWG7 10499348 IC50 = 2000 nM T83813 C6TQV3 10501785 IC50 = 240 nM T83813 CQE8U0 10502452 IC50 = 467735.14 nM T83813 CQA0U8 10503674 Ki = 25.12 nM T83813 CJC3R6 10504100 IC50 = 1500 nM T83813 C1FV7A 10516340 IC50 = 239.88 nM T83813 C28FSI 10517019 Ki = 316.23 nM T83813 CQD7L4 10518435 Ki = 5.012 nM T83813 CTP65K 10519608 IC50 = 13803.84 nM T83813 CUQ03E 10520440 Ki = 19 nM T83813 COTM08 10520537 Ki = 31.62 nM T83813 C8WR5O 10522029 IC50 = 2000 nM T83813 C2B9PT 10522146 Ki = 48 nM T83813 C7M0YQ 10523090 IC50 = 102329.3 nM T83813 CL1R5C 10523100 Ki = 25.12 nM T83813 C90TWP 10524876 IC50 = 320 nM T83813 CNE54K 10526362 IC50 = 1000000 nM T83813 CTO2C7 10526501 Ki = 25.12 nM T83813 CRK20I 10526616 Ki = 1.259 nM T83813 CNU6K9 10527432 Ki = 10 nM T83813 C4EN0P 10528314 Ki = 3.162 nM T83813 C3BXP0 10538127 Ki = 12.59 nM T83813 CYKP58 10539093 IC50 = 57543.99 nM T83813 CKG7E2 10541003 Ki = 4190 nM T83813 CTCN20 10543551 Ki = 25.12 nM T83813 C7M4CX 10544858 Ki = 363.08 nM T83813 CT80DS 10546033 Ki = 2.512 nM T83813 C48BRW 10546334 Ki = 64.57 nM T83813 CFN8B5 10546440 IC50 = 13803.84 nM T83813 CJ2T5R 10547091 IC50 = 300 nM T83813 CTLF72 10547809 IC50 > 100000 nM T83813 C1LV7P 10548259 IC50 = 13489.63 nM T83813 CMGY61 10549658 Ki = 5.012 nM T83813 CBU41F 10550405 Ki = 1 nM T83813 C0PV1R 10550406 Ki = 5.012 nM T83813 CE59TG 10553922 IC50 > 100000 nM T83813 CUZ2O8 10560133 Ki = 794.33 nM T83813 CNB05O 10566712 Ki = 25 nM T83813 CMV56C 10567817 Ki = 3.981 nM T83813 C5JY4K 10568666 IC50 > 100000 nM T83813 CW6VX8 10568745 IC50 = 10000 nM T83813 C2A6FZ 10568771 Ki = 0.3 nM T83813 CART26 10569395 IC50 = 36307.81 nM T83813 C7N1FY 10569470 IC50 = 61659.5 nM T83813 CBI9M2 10569827 Ki = 125.89 nM T83813 C9GSI8 10571450 IC50 > 100000 nM T83813 C8MSP1 10572269 Ki = 12.59 nM T83813 CY05PE 10573164 IC50 = 5888.44 nM T83813 C8O0ZN 10573656 Ki = 1.995 nM T83813 C9NQK8 10573762 Ki = 15.85 nM T83813 CHE80N 10573876 Ki < 5011.87 nM T83813 C4WGZ3 10574607 Ki = 3.162 nM T83813 C61SEA 10576618 IC50 = 1071.52 nM T83813 C8N7ML 10583453 Ki > 10000 nM T83813 CX8P3I 10583785 Ki = 15.85 nM T83813 CYH32C 10583942 EC50 = 72.3 nM T83813 CW71RC 10586264 Ki = 1 nM T83813 CH30OA 10589099 Ki = 316.23 nM T83813 C69LZJ 10590206 IC50 = 169.82 nM T83813 C0DX7G 10590360 IC50 = 346.74 nM T83813 COM18Y 10590891 Ki = 794 nM T83813 CY70EQ 10590892 Ki = 7.9 nM T83813 C9MUB5 10592633 Ki = 15.85 nM T83813 C4VLW7 10592646 Ki = 7.9 nM T83813 CH20WS 10593918 Ki = 25.12 nM T83813 CR1K9O 10594859 Ki = 316.23 nM T83813 CYNZ23 10595858 Ki = 3.162 nM T83813 C1SG9O 10597019 Ki < 10000 nM T83813 CO23YX 10597140 Ki < 10000 nM T83813 CW3TN5 10598044 IC50 = 19054.61 nM T83813 C2O3BC 10599545 Ki = 5.012 nM T83813 CAG6B7 10609802 Ki = 61.5 nM T83813 C74NSJ 10615016 Ki = 500 nM T83813 CRY9Q0 10617292 IC50 = 2454.71 nM T83813 COM89J 10617682 Ki = 12.59 nM T83813 C39FNQ 10619583 IC50 = 44668.36 nM T83813 C86KEZ 10620679 IC50 > 100000 nM T83813 CQH1X3 10621131 IC50 = 154.88 nM T83813 CMV72H 10622257 IC50 = 2630.27 nM T83813 CHD92F 10622347 Ki = 1949.84 nM T83813 CVKA91 10622480 Ki = 1.585 nM T83813 CW8YO5 10623020 Ki = 0.3162 nM T83813 CYT8G2 10623205 Ki = 0.631 nM T83813 CLCV43 10631592 Ki = 7.943 nM T83813 C01MLV 10637485 IC50 = 371.54 nM T83813 C8C2GN 10640055 Ki = 154 nM T83813 CSY57V 10641013 Ki = 6.31 nM T83813 C1A6ZO 10644514 IC50 = 560 nM T83813 C9XE8T 10645076 IC50 = 60 nM T83813 CCS31Z 10645335 IC50 > 100000 nM T83813 CH25VP 10645469 Ki = 3981.07 nM T83813 CQD6R2 10645615 IC50 = 851.14 nM T83813 CABG89 10646133 Ki = 0.631 nM T83813 CE6C0M 10660479 Ki = 79.43 nM T83813 C07AKO 10663820 IC50 > 100000 nM T83813 CZN9V7 10665419 IC50 = 2187.76 nM T83813 C4PV2W 10666301 IC50 = 5248.07 nM T83813 CB3C9Z 10667071 IC50 > 100000 nM T83813 C38YWE 10670191 Ki = 0.3981 nM T83813 CJC59K 10670813 Ki = 0.631 nM T83813 CGLN06 10679270 Ki > 10000 nM T83813 C65EDZ 10683685 Ki = 501.19 nM T83813 CVFC05 10686395 Ki = 15.85 nM T83813 C9ME8Z 10687130 Ki = 6.31 nM T83813 CC2I3O 10687827 Ki = 39.81 nM T83813 CTS4A1 10687868 IC50 > 100000 nM T83813 CP45QK 10689339 IC50 = 72443.6 nM T83813 C7BJO5 10690185 Ki = 3.162 nM T83813 C6YXC1 10691383 IC50 = 99 nM T83813 C3W5ZI 10693017 Ki < 10000 nM T83813 CJ04GI 10693836 Ki = 398.11 nM T83813 C7QZO5 10693974 Ki = 6.31 nM T83813 CW5K0A 10702890 Ki = 6190 nM T83813 CH4X8E 10704473 Ki = 1.259 nM T83813 C7XQN2 10705346 Ki = 12.59 nM T83813 C49IUL 10708935 Ki = 19 nM T83813 CML1J4 10709843 Ki = 31.62 nM T83813 CE8FX4 10709844 Ki = 50.12 nM T83813 C05JLO 10710246 Ki < 10000 nM T83813 C0Y1JL 10710785 Ki = 63.1 nM T83813 C9FAP1 10714457 IC50 = 10715.19 nM T83813 CIBU90 10714509 IC50 > 100000 nM T83813 C2SZA0 10714718 Ki = 25 nM T83813 CY3MJ1 10714852 Ki = 6.31 nM T83813 CJXI80 10715378 Ki = 1202.26 nM T83813 CVS29F 10715484 IC50 > 100000 nM T83813 CX8K5B 10717072 IC50 > 10000 nM T83813 C5NQX4 10717512 IC50 = 1071.52 nM T83813 CJR6Y5 10718089 Ki = 0.5012 nM T83813 CWV5A9 10718277 IC50 = 800 nM T83813 CVK2T3 10718731 IC50 = 281838.29 nM T83813 CM7N9Q 10719857 IC50 = 15488.17 nM T83813 CIL87B 10728235 IC50 = 424 nM T83813 CI0GE8 10737848 IC50 = 8317.64 nM T83813 CY1M6L 10738329 IC50 = 5248.07 nM T83813 CJH65T 10738619 Ki = 31.62 nM T83813 C1ZH6B 10739272 IC50 = 2570.4 nM T83813 C9F8CO 10739725 Ki = 3.162 nM T83813 CM3ZH1 10740447 Ki = 19.95 nM T83813 CQ95BN 10740494 Ki = 0.7943 nM T83813 CE5U6G 10740495 Ki = 5.012 nM T83813 C49CTY 10741816 Ki = 2.512 nM T83813 C7H8VX 10751567 Ki = 118.3 nM T83813 CZO1E3 10753377 IC50 = 269.15 nM T83813 C17OFU 10756517 IC50 = 758.58 nM T83813 CPQ40M 10759541 IC50 = 90 nM T83813 C85XRC 10762125 Ki = 19.95 nM T83813 CAO80C 10762881 Ki = 2500 nM T83813 CBUA63 10764263 Ki = 0.631 nM T83813 CQ4X1W 10766449 Ki = 0.631 nM T83813 C26JIN 10767350 Ki = 2.512 nM T83813 CIQ1E3 10774565 Ki = 125.89 nM T83813 C5PC0L 10774796 Ki = 3.981 nM T83813 C3SB0F 10776565 Ki = 3.981 nM T83813 CWSA98 10777682 IC50 = 41686.94 nM T83813 CX0B6M 10781655 Ki = 19.95 nM T83813 CG9MZ2 10784967 Ki = 50.12 nM T83813 C6ISL1 10788207 IC50 = 360 nM T83813 C5H1DA 10789000 IC50 = 11000 nM T83813 COJ20B 10790813 IC50 = 213796.21 nM T83813 CF2R3P 10791286 Ki = 1.995 nM T83813 C8ETQ1 10800216 Ki = 100 nM T83813 CC7J3N 10803066 Ki = 39.81 nM T83813 CVR74P 10803240 Ki = 10 nM T83813 C6LFB4 10804909 Ki = 3388.44 nM T83813 CO85JI 10804995 Ki = 229.09 nM T83813 CFH1Q4 10805130 Ki = 85 nM T83813 C4VA1L 10805623 IC50 = 10000 nM T83813 C8S4PF 10808909 IC50 = 1380384.26 nM T83813 CG5B6Z 10808965 Ki = 3.162 nM T83813 C31KNV 10809188 Ki = 81.28 nM T83813 C4K3SY 10809561 IC50 = 154881.66 nM T83813 C5J4ND 10809876 IC50 = 1200 nM T83813 C6BE4R 10810641 Ki < 10000 nM T83813 CT65RQ 10811153 Ki = 3.981 nM T83813 CQN8A4 10811876 IC50 = 3890.45 nM T83813 CUD58N 10812577 Ki = 1995.26 nM T83813 CKU7G0 10813396 Ki = 79.43 nM T83813 CCWH19 10814515 IC50 = 23442.29 nM T83813 CU06IQ 10823155 Ki = 1.259 nM T83813 CT1I7H 10826076 IC50 = 354.81 nM T83813 CF3N5R 10826203 IC50 = 100 nM T83813 CPXC32 10830245 Ki = 19.95 nM T83813 CCN0A5 10830746 Ki = 10 nM T83813 C5J1HW 10832055 IC50 = 520 nM T83813 CN0Z9Y 10833258 IC50 = 707.95 nM T83813 CL0BO9 10834414 IC50 > 100000 nM T83813 C8MHZ9 10835110 Ki < 1000 nM T83813 C5AI2P 10835537 Ki = 5.012 nM T83813 CFE3J6 10835585 Ki = 6.31 nM T83813 CGX81B 10837002 Ki = 0.631 nM T83813 CL3XI5 10837468 Ki = 0.5012 nM T83813 CDOH18 10851309 Ki > 2000 nM T83813 CIQS30 10852612 IC50 = 354.81 nM T83813 C1R3OJ 10852828 Ki = 125.89 nM T83813 C0VQ3C 10853014 Ki = 5 nM T83813 CBD60Q 10853821 IC50 > 100000 nM T83813 C62ZSF 10854005 Ki = 3.981 nM T83813 CV6ZN3 10861900 Ki = 39 nM T83813 C20CTE 10873003 Ki = 28 nM T83813 CVT7J1 10873805 Ki = 144 nM T83813 C9OH3F 10881914 Ki < 10000 nM T83813 CCJ9Y2 10898996 EC50 = 634 nM T83813 CX65PW 10907460 IC50 = 1420 nM T83813 C2BZ9X 10912292 IC50 > 10000 nM T83813 C2UZ8H 10917953 Ki = 410 nM T83813 CDR7G5 10925892 Ki = 320 nM T83813 C9T7LS 10926165 Ki = 281.84 nM T83813 C9OI8S 10927262 Ki = 39 nM T83813 CT79NZ 10927276 IC50 = 345 nM T83813 CM0OS2 10939174 IC50 = 1830 nM T83813 C4PK7X 10971209 Ki = 41 nM T83813 C5NRU3 10973768 Ki = 1100 nM T83813 C51NOQ 10982183 Ki = 20.42 nM T83813 CK6VF7 10991109 Ki = 493 nM T83813 C0BUR1 10991521 Ki = 450 nM T83813 C4O7MD 10994400 Ki = 28.6 nM T83813 CJC9K4 11005810 IC50 = 2760 nM T83813 CE6HJ8 11013863 Ki = 440 nM T83813 C6GT4A 11014340 Ki = 104.71 nM T83813 C3FIP5 11016205 Ki = 35.5 nM T83813 CH9GU5 11016418 Ki > 4200 nM T83813 C4T8LY 11020695 Ki = 20 nM T83813 CV6S3D 11023903 Ki < 10000 nM T83813 CS0Z2D 11024311 Ki < 10000 nM T83813 CG9JC8 11036563 Ki = 47 nM T83813 C6EBF3 11048769 IC50 = 652 nM T83813 CG41BK 11071079 IC50 = 3450 nM T83813 CUJ4W7 11071135 Ki > 4200 nM T83813 CGEY62 11079151 Ki = 1500 nM T83813 CM2BD4 11092112 Ki > 4200 nM T83813 C76FKX 11100514 Ki = 600 nM T83813 CSZ9C6 11121409 Ki = 1698.24 nM T83813 C6ASW7 11128034 EC50 = 158 nM T83813 CHX96W 11133309 Ki = 18 nM T83813 CJL04G 11141324 Ki = 851.14 nM T83813 CHEV46 11148641 EC50 = 330 nM T83813 CZK0E6 11150514 Ki = 1100 nM T83813 CTHA45 11151653 EC50 = 8 nM T83813 C5HEF8 11154832 Ki = 15.85 nM T83813 C3NH7G 11160564 EC50 = 19.95 nM T83813 C4SOG5 11163458 Ki = 48 nM T83813 CW7Y9O 11163741 Ki = 31.62 nM T83813 C8ZN3B 11166042 IC50 = 9665 nM T83813 CK23LI 11166827 Ki = 1.995 nM T83813 C1SXY8 11171464 EC50 = 2.512 nM T83813 COG98Y 11171955 EC50 = 56 nM T83813 CLP45Z 11175045 Ki = 51 nM T83813 C6OLX8 11176570 EC50 = 18 nM T83813 C5TR6Q 11178237 Ki = 251.19 nM T83813 C6CL1Y 11178830 Ki = 2511.89 nM T83813 C4FYN6 11185858 Ki = 321 nM T83813 C0W4SM 11186523 Ki = 1.5 nM T83813 CDA9Z8 11187156 Ki = 57 nM T83813 C90ZAQ 11195293 EC50 = 1358 nM T83813 C9N5QU 11200511 Ki = 289 nM T83813 CPS26T 11201645 IC50 > 10000 nM T83813 C52BGU 11206703 EC50 = 3 nM T83813 CPX23W 11209208 IC50 > 10000 nM T83813 C5NA0Z 11209786 EC50 = 14 nM T83813 C2A1PL 11221167 Ki = 7 nM T83813 CAF7T3 11222829 Ki = 1428 nM T83813 C6D1MZ 11223004 Ki = 566 nM T83813 CJS0I7 11225281 Ki = 3.162 nM T83813 CZFH27 11231392 EC50 = 107 nM T83813 CXB4Q8 11233293 Ki = 34 nM T83813 CNR71Z 11235362 Ki = 19.95 nM T83813 CBO29U 11236301 Ki = 1.995 nM T83813 C2JOS6 11237290 Ki = 0.7943 nM T83813 C9HB3Z 11247569 Ki = 10 nM T83813 C90WSG 11248705 Ki = 3981.07 nM T83813 C3XS7W 11253485 EC50 = 514 nM T83813 C6DA3J 11258838 Ki = 63.1 nM T83813 CWD43K 11264345 EC50 = 19.95 nM T83813 C2U7OP 11270012 IC50 = 55000 nM T83813 C4S2VF 11277147 Ki > 1000 nM T83813 C27GXZ 11277680 IC50 > 10000 nM T83813 CIG85H 11282247 IC50 > 33000 nM T83813 CLFM61 11282335 Ki = 5.012 nM T83813 C28ZWI 11283484 Ki = 125.89 nM T83813 CJD16T 11288140 EC50 = 281 nM T83813 COQ7H8 11290492 Ki = 133 nM T83813 C83DSZ 11292350 Ki = 2.512 nM T83813 C08UHY 11294575 Ki = 3.981 nM T83813 C57GTA 11299968 IC50 > 10000 nM T83813 CM43ZJ 11300712 EC50 = 12 nM T83813 CB0UJ7 11302765 EC50 = 16 nM T83813 C9BLC7 11304596 Ki > 5011.87 nM T83813 CU4L6M 11304816 IC50 = 970 nM T83813 CJS9C0 11304851 IC50 > 10000 nM T83813 C49LMW 11305844 Ki = 0.3981 nM T83813 CI79LV 11307899 Ki = 15.85 nM T83813 CUXZ91 11311148 IC50 > 10000 nM T83813 C2GZD3 11311204 IC50 > 10000 nM T83813 CLQM72 11312820 Ki = 369 nM T83813 CU81GW 11313985 EC50 = 3 nM T83813 C1EAK6 11324968 EC50 = 55 nM T83813 C46TGM 11328372 Ki = 10 nM T83813 CZ8R4L 11328744 Ki = 10 nM T83813 C2DVE9 11333043 EC50 = 794.33 nM T83813 CV1I4W 11336079 Ki = 332 nM T83813 CDN79K 11346775 EC50 = 86 nM T83813 CHW9G0 11347858 Ki = 460 nM T83813 CJT5E1 11350623 Ki = 155 nM T83813 CU5L7F 11361103 Ki = 456 nM T83813 C6D1WP 11363880 Ki = 63.1 nM T83813 CDOP76 11374796 Ki = 3.981 nM T83813 CBV52J 11384146 Ki = 231 nM T83813 CF4OX6 11397149 Ki > 10000 nM T83813 C7IPE2 11400855 EC50 = 909 nM T83813 C6ZXH8 11412671 Ki = 3170 nM T83813 C0UWG6 11413558 Ki = 826 nM T83813 C7RAB8 11414184 Ki = 19 nM T83813 COZJ91 11416698 EC50 = 241 nM T83813 CFX98O 11418182 Ki = 69 nM T83813 CNM62W 11419526 Ki = 1 nM T83813 CIB9K8 11427139 Ki = 43 nM T83813 C7BZA8 11429246 Ki = 10 nM T83813 C3K7TG 11430311 Ki = 1.259 nM T83813 C4LWN6 11431347 Ki = 25.12 nM T83813 CYZC62 11437171 Ki = 40 nM T83813 CF94ZE 11447552 EC50 = 6 nM T83813 CY06IJ 11448649 Ki = 20 nM T83813 CHG7Q4 11453346 Ki = 15.85 nM T83813 CHS2R7 11453704 Ki = 2.512 nM T83813 C1W8QL 11454107 Ki = 6.31 nM T83813 CY76VX 11463745 Ki = 3.981 nM T83813 CDTI21 11465413 Ki = 1.995 nM T83813 C1QL6G 11475519 Ki = 1.585 nM T83813 CB2X1C 11483068 EC50 = 49 nM T83813 CJ6GV8 11492300 EC50 = 43 nM T83813 CSP63L 11493484 EC50 = 4.3 nM T83813 C8FN2P 11494093 Ki > 1000 nM T83813 C6L8DU 11495754 IC50 = 5900 nM T83813 C9YME5 11496313 IC50 > 10000 nM T83813 C0AG7D 11497283 Ki = 12.4 nM T83813 CFY18U 11499800 EC50 = 20 nM T83813 CASD80 11501253 Ki > 1000 nM T83813 C16AXW 11501537 Ki > 1000 nM T83813 CYC7D5 11503034 Ki > 1000 nM T83813 CXG04S 11503810 Ki = 5900 nM T83813 CJ2O6D 11514226 EC50 = 1.1 nM T83813 C1TC0B 11517754 Ki = 1150 nM T83813 CT6O8G 11519011 Ki = 3.162 nM T83813 C9S7ZD 11519589 Ki = 251.19 nM T83813 C38QFE 11530118 IC50 > 10000 nM T83813 C4HI2Q 11531833 Ki = 398.11 nM T83813 CTA58E 11531941 Ki > 10000 nM T83813 C7DBO0 11537385 Ki > 1000 nM T83813 CQ08DH 11539632 IC50 = 2500 nM T83813 CX0DJ3 11545423 Ki = 47 nM T83813 C5ZY6N 11545813 Ki = 3513 nM T83813 C9VC7O 11551780 IC50 > 10000 nM T83813 CC4J3M 11553617 Ki > 10000 nM T83813 C1V5CH 11559090 Ki > 10000 nM T83813 C59SVL 11563383 IC50 = 4700 nM T83813 CVP1Q9 11567578 Ki = 169 nM T83813 CD3Z7J 11567928 Ki = 190 nM T83813 C3DU6B 11567937 Ki = 39.81 nM T83813 CNH1K4 11568826 Ki > 10 nM T83813 C8NMI4 11575479 Ki > 10000 nM T83813 C4HS8T 11577304 Ki = 794.33 nM T83813 CMTN14 11579853 EC50 = 12 nM T83813 C6JC2T 11580039 IC50 > 10000 nM T83813 CPA3J7 11583744 IC50 = 4000 nM T83813 C6D1MA 11584660 Ki > 3981.07 nM T83813 C90XFB 11587397 EC50 = 30 nM T83813 C4OK0R 11588889 Ki = 398.11 nM T83813 C1M2CP 11589069 Ki = 690 nM T83813 C5TQ3Y 11595191 EC50 = 41 nM T83813 CU45DK 11595209 Ki > 10000 nM T83813 CGX8F6 11596869 Ki > 7870000 nM T83813 C6G7WS 11603119 Ki = 43 nM T83813 CGD62Y 11603486 Ki = 1350 nM T83813 C1D5YN 11604671 Ki = 25.12 nM T83813 CZ2OG1 11608308 EC50 = 3 nM T83813 CYF3M8 11609026 EC50 = 3.3 nM T83813 CL51UW 11612277 Ki = 1140 nM T83813 C5JZ6R 11615459 EC50 = 45 nM T83813 CR6S3I 11624518 Ki = 8440 nM T83813 C4YG6K 11625339 Ki = 25.12 nM T83813 CB7M8E 11625642 Ki = 173 nM T83813 CDQ02B 11627746 Ki = 1.6 nM T83813 CN3WL4 11630147 Ki = 19 nM T83813 C9F4UK 11630623 EC50 = 11 nM T83813 CX36IC 11634230 IC50 = 18000 nM T83813 C2OU7Y 11638332 Ki > 10000 nM T83813 C19UMY 11638640 Ki > 1000 nM T83813 CH89AK 11639248 Ki > 1000 nM T83813 C9OXY8 11644842 EC50 = 59 nM T83813 C5A4YW 11648240 IC50 = 5700 nM T83813 CVU40P 11652359 EC50 = 82 nM T83813 CM57PQ 11652452 EC50 = 3.3 nM T83813 C1HDM5 11653679 Ki = 1425 nM T83813 CPH9X5 11655664 Ki > 10000 nM T83813 CRES94 11656729 Ki = 31.62 nM T83813 C4L7TV 11662592 Ki = 5.5 nM T83813 CR7WX0 11665991 Ki = 1547 nM T83813 CI81RY 11666237 EC50 = 17 nM T83813 CAI7R5 11673842 EC50 = 218 nM T83813 C7SNQ8 11675550 Ki = 316.23 nM T83813 C4KUL7 11676638 Ki = 22 nM T83813 CMQX39 11676873 Ki = 326 nM T83813 CYC89S 11680606 Ki = 450 nM T83813 CQZ89L 11684204 Ki = 15.85 nM T83813 CEQ6W7 11694810 Ki = 390 nM T83813 CCE9H2 11695000 EC50 = 1 nM T83813 CDV58J 11696813 Ki = 206 nM T83813 C65TAC 11698513 Ki = 120 nM T83813 CI1LY5 11698617 Ki > 10000 nM T83813 CU8QZ9 11701315 EC50 = 34 nM T83813 CN7Q5B 11710154 Ki = 158.49 nM T83813 CRH96P 11716185 EC50 = 26 nM T83813 CV9G1F 11719283 Ki = 3.981 nM T83813 CB3AM8 11719524 Ki = 225 nM T83813 CF3EA1 11719622 Ki = 2.512 nM T83813 CAF0J1 11725183 IC50 = 794.33 nM T83813 C2ML7T 11725312 IC50 = 794.33 nM T83813 CLYJ75 11729823 Ki = 16.6 nM T83813 C7PVL8 11730467 IC50 = 4070 nM T83813 C5MET7 11736340 EC50 = 1260 nM T83813 C53KHL 11737032 Ki = 31 nM T83813 CH0PB9 11737939 EC50 = 20 nM T83813 C05TYZ 11739217 EC50 = 63 nM T83813 C57IKL 11740526 Ki < 1000 nM T83813 C8Q4ET 11742218 Ki = 1.995 nM T83813 CPG15O 11743399 IC50 > 1000 nM T83813 CUE3K5 11749963 Ki = 50.12 nM T83813 C6SKL1 11750162 Ki = 3.162 nM T83813 CK4LU1 11750342 Ki = 25.12 nM T83813 C45RXA 11750471 Ki = 31.62 nM T83813 CT7YB5 11753781 Ki = 6.31 nM T83813 C16EAQ 11760018 Ki = 575.44 nM T83813 C7KD9Z 11766873 Ki = 10 nM T83813 C43JMK 11774776 Ki = 125.89 nM T83813 CNZV46 11774955 Ki = 15.85 nM T83813 C4IQ8G 11775262 Ki = 1.585 nM T83813 CUT31Z 11777150 EC50 = 3 nM T83813 C4KNX5 11777180 IC50 = 1258.93 nM T83813 C2T3OV 11777228 IC50 = 3162.28 nM T83813 CM9A7S 11777810 IC50 = 1000 nM T83813 C0CZ2S 11783381 Ki = 190 nM T83813 CU5G2Q 11785555 Ki = 158.49 nM T83813 CGI2R8 11792032 IC50 = 11748.98 nM T83813 C09ECB 11792056 Ki = 50.12 nM T83813 CYR2L7 11793287 IC50 = 7413.1 nM T83813 CGVY61 11794853 IC50 = 457.09 nM T83813 CLEW30 11795165 Ki = 69.18 nM T83813 C8AWF3 11796209 IC50 = 8709.64 nM T83813 C90MLE 11797241 IC50 > 100000 nM T83813 C1M3BY 11797762 IC50 > 100000 nM T83813 CQ98FK 11819486 Ki = 21.3 nM T83813 CE6J4U 11820166 Ki = 11.8 nM T83813 COB43E 11825520 Ki = 58 nM T83813 CQ64OY 11949706 EC50 = 1 nM T83813 CP79ZF 11949710 Ki = 1.5 nM T83813 CEYG15 11949712 EC50 = 0.1 nM T83813 CWG8D2 11952353 EC50 = 1.4 nM T83813 C8JQL7 11957735 IC50 > 10000 nM T83813 CR7IZ8 11983273 EC50 = 103 nM T83813 CID7H8 12017581 Ki > 1000 nM T83813 CUD9A3 12017598 Ki = 5.012 nM T83813 CM95EO 12017599 Ki = 3.162 nM T83813 C8EDN0 12088080 Ki > 1000 nM T83813 C8RB6W 12088082 Ki = 160 nM T83813 C4CE8D 12111141 Ki = 10 nM T83813 CL29RB 12197243 Ki = 9 nM T83813 CTMH07 12370465 EC50 = 13 nM T83813 CM8FI1 12370466 EC50 = 3019 nM T83813 CHS34O 12440702 Ki = 8320 nM T83813 CNTW70 12763911 EC50 = 1995 nM T83813 C28QEX 12765746 Ki = 2.9 nM T83813 C6I4GL 12901777 Ki = 630 nM T83813 C2S1KL 12986493 Ki = 66 nM T83813 C8EXN6 12986494 Ki = 1 nM T83813 CU7CQ9 12986495 Ki = 7 nM T83813 CW65EI 12986496 Ki = 8 nM T83813 CVOX89 12986497 Ki = 516 nM T83813 C4EBZ6 12986498 Ki = 34 nM T83813 C2V9FL 13091268 Ki = 872.1 nM T83813 C2VAE5 13091273 Ki > 10000 nM T83813 CDK0W1 13385712 IC50 = 5110 nM T83813 CPFQ95 13764011 EC50 = 4.266 nM T83813 C9I7FG 14515722 Ki > 300000 nM T83813 CBG32N 14515723 Ki = 300000 nM T83813 CGW8C5 14515724 Ki = 100000 nM T83813 C5TU0D 14515725 EC50 = 416.87 nM T83813 C7IXM0 14515726 EC50 = 12000 nM T83813 CHIN31 14515727 Ki > 300000 nM T83813 CO8SN6 14515728 Ki > 300000 nM T83813 C4XL7T 14595518 Ki = 450 nM T83813 CJ16HE 15011385 Ki = 16 nM T83813 C7VAI1 15011772 IC50 > 10000 nM T83813 CN0KL5 15021875 Ki = 2818.38 nM T83813 C5F7NM 15021876 Ki = 234.42 nM T83813 CK21HZ 15226949 IC50 = 34.67 nM T83813 CTX2Z7 15233110 IC50 > 1000 nM T83813 C30CHU 15512229 Ki < 316.23 nM T83813 C5ZK0U 15640062 EC50 = 63.1 nM T83813 C6US3O 15711850 Ki = 58.4 nM T83813 C5PO3N 15711869 Ki = 200 nM T83813 CL50KS 15983730 Ki > 10000 nM T83813 CCY53Q 15984073 EC50 = 6 nM T83813 C1LWZ6 16006605 Ki = 74 nM T83813 CK36NS 16006607 Ki = 488 nM T83813 COUI94 16022762 IC50 > 10000 nM T83813 CD65KI 16046157 IC50 > 100000 nM T83813 C37FIP 16047544 EC50 = 1.3 nM T83813 C6OYT5 16062136 Ki = 100 nM T83813 CBWZ28 16062137 Ki = 400 nM T83813 CLG47H 16062139 Ki = 1020 nM T83813 C6Y3LW 16062143 Ki = 410 nM T83813 C0K1DQ 16062145 Ki = 5000 nM T83813 C9HQ7A 16062266 Ki = 1000 nM T83813 CM45DK 16062270 Ki = 110 nM T83813 C09LXV 16062651 Ki = 1000 nM T83813 C8PU1B 16062781 Ki = 200 nM T83813 CCL8Z7 16062782 Ki = 23 nM T83813 C7VW3X 16062783 Ki = 120 nM T83813 CXQ0L4 16062784 Ki = 460 nM T83813 CKB71R 16062785 Ki = 80 nM T83813 CPS49Q 16062788 Ki = 20 nM T83813 C4AZV6 16062910 Ki = 15 nM T83813 CK08NX 16062911 Ki = 38 nM T83813 C4JTB1 16062912 Ki = 50 nM T83813 CQBU41 16063039 Ki = 150 nM T83813 C16OJN 16063047 Ki = 5000 nM T83813 C51YGX 16063181 Ki = 75 nM T83813 C1SR0O 16071847 Ki = 573 nM T83813 CD3E8L 16093484 Ki = 26 nM T83813 CEW91O 16093485 Ki = 19 nM T83813 CQS4V1 16112801 IC50 = 1127 nM T83813 CEWI25 16115148 Ki = 1030 nM T83813 CA15XJ 16115267 EC50 = 18 nM T83813 CVL4O8 16115269 Ki = 74 nM T83813 CA15YJ 16115271 EC50 = 10 nM T83813 CU86YM 16115381 EC50 = 28 nM T83813 CCZ1E8 16115388 Ki = 335 nM T83813 C3PE9N 16115390 Ki = 5060 nM T83813 C8KMO4 16115392 EC50 = 54 nM T83813 CIN2U9 16115511 EC50 = 46 nM T83813 CJ1YO5 16115513 EC50 = 5 nM T83813 C5RK9P 16115515 EC50 = 35 nM T83813 C4J7OR 16115517 EC50 = 1.4 nM T83813 CVF2A4 16115521 EC50 = 246 nM T83813 CJO13N 16115644 EC50 = 17 nM T83813 CXNA76 16115647 Ki = 1610 nM T83813 C0F5WY 16115650 Ki = 900 nM T83813 C4IT3C 16115652 EC50 = 11 nM T83813 CWG94S 16115654 EC50 = 6 nM T83813 CZ1WJ4 16117151 Ki = 2427 nM T83813 CM32ZX 16117153 Ki > 5000 nM T83813 CXTB90 16117279 Ki = 1767 nM T83813 C1F2LS 16118795 Ki > 5000 nM T83813 C69VDS 16118923 Ki > 5000 nM T83813 C9EF6M 16215237 Ki = 2.512 nM T83813 C4YJD2 16456446 IC50 = 1085 nM T83813 CB7Y4I 16456451 IC50 = 7.8 nM T83813 C97FJS 16456452 IC50 = 5422 nM T83813 CM0H6S 16456546 IC50 > 10000 nM T83813 C0JU4P 16456618 IC50 > 10000 nM T83813 CQR85B 16456712 IC50 = 8491 nM T83813 C7ZMA0 16456728 IC50 = 1179 nM T83813 C9K2VJ 16456770 IC50 > 10000 nM T83813 CU7I8O 16456771 IC50 = 7787 nM T83813 CL9O8C 16456772 IC50 > 10000 nM T83813 CI3O8J 16456776 IC50 > 10000 nM T83813 CM6K7Z 16456777 IC50 > 10000 nM T83813 CHY67G 16456778 IC50 = 5713 nM T83813 CKO26C 16456779 IC50 = 5833 nM T83813 CN6UT8 16456781 IC50 > 10000 nM T83813 CE0JF9 16456782 IC50 > 10000 nM T83813 CEF9Y6 16456783 IC50 > 10000 nM T83813 CWJ5H0 16456784 IC50 = 3306 nM T83813 CR78LC 16456786 IC50 = 2071 nM T83813 CU3FX5 16456787 IC50 = 1500 nM T83813 CK7MR1 16456789 IC50 = 20.1 nM T83813 C8C1OK 16456790 IC50 = 494 nM T83813 CEA84P 16456791 IC50 = 836 nM T83813 CNS7G3 16456792 IC50 = 416 nM T83813 CTPG46 16456794 IC50 = 148 nM T83813 CHP1W2 16456795 IC50 = 1725 nM T83813 C72BAI 16659061 Ki > 100000 nM T83813 C23NUI 16659197 IC50 > 100000 nM T83813 CZ2IS9 16660294 Ki > 10000 nM T83813 CB7G3R 16718920 IC50 > 1000 nM T83813 C6DS7K 16739334 Ki = 65 nM T83813 CHA74P 16743289 EC50 = 0.2 nM T83813 CNOW10 17095595 IC50 > 10000 nM T83813 C1GR9B 17954204 EC50 = 12 nM T83813 C9WUR7 17956720 Ki = 15.85 nM T83813 C3J2EH 17989823 Ki = 1.585 nM T83813 CV7T6Z 17989828 Ki = 10 nM T83813 CZO18R 17989871 Ki = 1.259 nM T83813 C8JEI2 17989875 Ki = 79.43 nM T83813 C9RY6L 18005120 Ki = 0.3981 nM T83813 C9PV8A 18180076 IC50 = 5147 nM T83813 CZ58PY 18357723 Ki = 15.85 nM T83813 C2I7CO 18357724 Ki = 7.943 nM T83813 CS90WO 18357730 Ki = 0.3981 nM T83813 CHXQ26 18366015 IC50 > 10000 nM T83813 C2DFS4 18435980 IC50 = 55 nM T83813 CCS6E4 18436055 IC50 = 630 nM T83813 C7MUE8 18436066 IC50 > 1000 nM T83813 C9HN3G 18436075 IC50 = 160 nM T83813 CA9UL8 18436082 IC50 = 240 nM T83813 CDQS35 18436083 IC50 = 280 nM T83813 C1WJ0Z 18436085 IC50 = 7.4 nM T83813 C3CYE7 18436094 IC50 = 78 nM T83813 CF7Q1R 18436112 IC50 > 1000 nM T83813 CS24AR 18436114 IC50 > 1000 nM T83813 C34WKZ 18436115 IC50 = 660 nM T83813 C0H7OP 18436117 IC50 = 540 nM T83813 C7X1SY 18436120 IC50 = 930 nM T83813 C9F2DA 18436123 IC50 = 830 nM T83813 CW6HU8 18436126 IC50 = 570 nM T83813 C82DBE 18475509 Ki = 50.12 nM T83813 C3DP7R 18475581 Ki = 630.96 nM T83813 CNP6Q1 18475610 Ki = 50.12 nM T83813 CHP8Q5 18475630 Ki = 79.43 nM T83813 C8EQN1 18475647 Ki = 31.62 nM T83813 CK0TX2 18516642 Ki = 3.162 nM T83813 CUZ6M7 18520432 EC50 = 0.7943 nM T83813 CL24WJ 18545468 Ki = 2540 nM T83813 CAP6L1 18672590 Ki = 158.49 nM T83813 CNAK30 18715554 Ki = 72 nM T83813 CSIT54 18715555 Ki = 16 nM T83813 CNFG32 18715558 Ki = 37 nM T83813 C03DXY 18715561 Ki = 27 nM T83813 CG2K0J 18715564 Ki = 2.4 nM T83813 C2ST7K 18735305 Ki = 17 nM T83813 CUC5V9 18735309 Ki = 26 nM T83813 C9GW5T 18735313 Ki = 13 nM T83813 CRLH78 18931123 Ki = 39.81 nM T83813 C42WCN 18931133 Ki = 10 nM T83813 CW7QF4 18931150 Ki = 6.31 nM T83813 CZKR20 18931163 Ki = 7.943 nM T83813 CW5GP0 18931172 Ki = 398.11 nM T83813 C7PU3Q 18931202 Ki = 3.981 nM T83813 C1INB0 18931217 Ki = 79.43 nM T83813 CY10RA 18931344 Ki = 31.62 nM T83813 CODQ12 18931348 Ki = 3.162 nM T83813 C37ZWN 18931357 Ki = 5.012 nM T83813 C5LQX3 18931377 Ki = 50.12 nM T83813 C5T4BW 18931420 Ki = 1.585 nM T83813 CY60VR 18931422 Ki = 0.1995 nM T83813 CQXS12 18986247 Ki = 1.995 nM T83813 CURH72 19036356 Ki = 3.162 nM T83813 C6MQ4P 19036360 Ki = 0.3981 nM T83813 CFB7P2 19036374 Ki = 3.981 nM T83813 CF0X7Z 19036377 Ki = 7.943 nM T83813 C9E0JS 19036385 Ki = 3.981 nM T83813 C48OSF 19036480 Ki = 5.012 nM T83813 C1HL8Z 19356259 Ki = 1.995 nM T83813 CCSX34 19390921 Ki > 10000 nM T83813 CJ6L5B 19426632 IC50 = 5.623 nM T83813 C6AOE8 19426635 IC50 = 7.079 nM T83813 CT1Q8M 19426644 IC50 = 16.22 nM T83813 CFYH89 19426650 IC50 = 691.83 nM T83813 C9ODM1 19426658 IC50 > 1000 nM T83813 CQ3JL0 19956256 IC50 = 2137.96 nM T83813 C7T8JC 19958494 Ki > 10000 nM T83813 C6LI5E 19958507 Ki > 10000 nM T83813 CLVT08 19978038 IC50 = 275.42 nM T83813 CF34NC 19978059 IC50 > 100000 nM T83813 C3M6OA 20026449 EC50 = 2951.21 nM T83813 CECV54 20098653 IC50 > 10000 nM T83813 C5Q6FW 20576921 Ki = 195 nM T83813 C4U8TE 20726100 Ki = 4.7 nM T83813 C71ZTU 20726102 Ki = 6.8 nM T83813 C5Z7FO 20726104 Ki = 64 nM T83813 CNJY54 20824945 Ki = 1.3 nM T83813 CSN4T5 20824946 Ki = 34 nM T83813 CRUI61 20824949 Ki = 680 nM T83813 CBY03N 20846175 Ki < 10000 nM T83813 C1Q3PH 20868365 IC50 > 10000 nM T83813 CTF21H 20917177 IC50 > 10000 nM T83813 CD6Q2A 20917185 IC50 > 10000 nM T83813 CAX9P3 20920181 IC50 > 10000 nM T83813 CYN83I 20924687 IC50 > 10000 nM T83813 C4YN8T 20924857 IC50 > 10000 nM T83813 C6U8JV 20925045 IC50 = 4169 nM T83813 CXZG31 20925636 IC50 > 10000 nM T83813 CYUT29 20926111 IC50 = 5294 nM T83813 C8YGH5 20940652 IC50 = 222 nM T83813 CPLT36 21044391 Ki = 54 nM T83813 C6JSC0 21044398 Ki = 39 nM T83813 CAO91K 21099378 Ki = 7 nM T83813 C9MDU4 21099413 Ki = 2700 nM T83813 C2LMD4 21099424 Ki = 526 nM T83813 CJB73F 21099433 Ki = 127 nM T83813 CQU60A 21099448 Ki > 4000 nM T83813 CBCL34 21099463 Ki = 43 nM T83813 C36INC 21099465 Ki = 410 nM T83813 C6GRC9 21099470 Ki = 25 nM T83813 CY75XP 21099472 Ki > 4000 nM T83813 CCO7D2 21099473 Ki > 4000 nM T83813 CP94VE 21099486 Ki = 21 nM T83813 CF90PJ 21099505 Ki = 41 nM T83813 CDBY94 21099514 Ki > 4000 nM T83813 CB12UT 21099515 Ki > 4000 nM T83813 CPWG76 21302447 Ki = 664 nM T83813 CQF01H 21302453 Ki = 672 nM T83813 CTFH75 21302454 Ki = 112 nM T83813 CGL9D3 21302455 Ki = 754 nM T83813 CY3M2Z 21302456 Ki = 259 nM T83813 CY6H3F 21302457 Ki = 258 nM T83813 CB4V8Q 21302458 Ki = 172 nM T83813 C9WD5O 21302459 Ki = 253 nM T83813 C7TSU2 21302471 Ki = 452 nM T83813 CWHT46 21302483 EC50 = 943 nM T83813 C7Y0HC 21302486 Ki = 280 nM T83813 CJP08R 21302487 Ki = 385 nM T83813 CB7S2R 21302488 Ki = 287 nM T83813 COD3H1 21302489 Ki = 498 nM T83813 C2EO0C 21302505 Ki = 259 nM T83813 C56MVN 21302580 Ki = 5.2 nM T83813 C3T5HF 21509921 Ki = 10 nM T83813 CQO1R3 21786603 Ki = 103 nM T83813 CSQ2Y0 22017550 Ki = 557 nM T83813 CBN84K 22065997 Ki > 10000 nM T83813 CQMS26 22292784 EC50 = 25.12 nM T83813 CC6AJ0 22368315 EC50 = 8 nM T83813 CEXB75 22517723 IC50 > 10000 nM T83813 CP97QA 22517837 IC50 = 9223 nM T83813 C5IE1F 22619858 Ki = 3.162 nM T83813 CD9M5W 22720253 Ki = 30 nM T83813 C9JN0F 22720399 Ki = 23 nM T83813 CB6JH2 22720609 Ki = 14 nM T83813 CJ86XR 23022422 IC50 = 760 nM T83813 C26ESM 23022499 IC50 = 310 nM T83813 CJS4U2 23022589 IC50 > 1000 nM T83813 C2VA8B 23139417 Ki = 398.11 nM T83813 C4OC9V 23360842 Ki = 391 nM T83813 C1RIA7 23395431 EC50 = 10 nM T83813 CA6QL5 23462894 Ki = 66 nM T83813 C0U2TC 23467920 EC50 > 10000 nM T83813 CX6L7J 23602561 IC50 > 10000 nM T83813 CMI12X 23604139 IC50 = 5627 nM T83813 CXD3E6 23625925 Ki = 123.03 nM T83813 CY78MC 23631023 Ki > 1000 nM T83813 C5V6KM 23631112 Ki > 1000 nM T83813 C0YM5F 23631117 Ki > 1000 nM T83813 CU1M2C 23631288 Ki > 1000 nM T83813 CQ1M3P 23631387 Ki > 1000 nM T83813 C4LEI9 23631388 Ki > 1000 nM T83813 CL4CF8 23642306 Ki = 707.95 nM T83813 C9U6TM 23642307 Ki = 165.96 nM T83813 CR1M4E 23652278 EC50 = 15.85 nM T83813 CG78OH 23658143 Ki > 10000 nM T83813 CY68EQ 23658144 Ki = 186.21 nM T83813 CBS59I 23658145 Ki > 10000 nM T83813 CLJ03E 23658146 Ki = 416.87 nM T83813 CNU2X4 23725134 IC50 > 1000 nM T83813 CZ4BW9 24044716 IC50 = 1010 nM T83813 C0I2HU 24769156 Ki > 1000 nM T83813 CD7CV6 24771120 Ki > 2000 nM T83813 CGX8K2 24773648 EC50 = 1258.93 nM T83813 CSCJ40 24773649 EC50 = 3.981 nM T83813 C6T5XP 24773650 EC50 = 50.12 nM T83813 CLR9M6 24773651 EC50 = 6.31 nM T83813 CMA8Q6 24773728 EC50 = 19.95 nM T83813 C4O2YA 24773809 EC50 = 7.943 nM T83813 C7IT2S 24773814 EC50 = 39.81 nM T83813 C2U8IH 24773816 EC50 = 7.943 nM T83813 CTK36B 24773894 EC50 = 230 nM T83813 CG1V5R 24773895 EC50 = 7.943 nM T83813 C9WV5A 24773897 EC50 = 3.981 nM T83813 C6IF2A 24773900 EC50 = 199.53 nM T83813 CNOE28 24773901 EC50 = 794.33 nM T83813 C8R9DY 24773978 EC50 = 199.53 nM T83813 CF2U4K 24773979 EC50 = 316.23 nM T83813 C2E8SA 24810866 Ki > 10000 nM T83813 C14FOH 24810867 Ki = 1410 nM T83813 CT53OY 24810870 Ki = 2120 nM T83813 C82ZEQ 24810973 Ki > 10000 nM T83813 C8GX1Z 24811073 Ki > 10000 nM T83813 CX17DO 24811076 Ki = 8600 nM T83813 C6A8SY 24811079 Ki = 5614 nM T83813 CSD96T 24811182 Ki > 10000 nM T83813 COQ5U2 24811184 Ki = 4146 nM T83813 CG0FJ6 24811298 Ki = 2750 nM T83813 CKCF54 24811301 Ki > 10000 nM T83813 C1CH9O 24811415 Ki = 3866 nM T83813 CG49QZ 24811418 Ki > 10000 nM T83813 CGKV62 24811420 Ki = 3573 nM T83813 CL71GM 24811748 Ki = 2933 nM T83813 CO6ZG1 24811751 Ki = 9800 nM T83813 C5IR4Z 24811854 Ki = 1420 nM T83813 C4CU8V 24811856 Ki > 10000 nM T83813 CO4ZF3 24811956 Ki > 10000 nM T83813 C7RY2Z 24811959 Ki = 2820 nM T83813 C6IY3J 24812067 Ki > 10000 nM T83813 CZL2H0 24812461 Ki > 10000 nM T83813 CUE6Q0 24812462 Ki > 10000 nM T83813 CB6D4T 24812467 Ki > 10000 nM T83813 CJN09A 24826786 Ki = 24 nM T83813 C3PQB2 24826787 EC50 = 16 nM T83813 CRKE01 24826788 EC50 = 22 nM T83813 C6BM3J 24826790 EC50 = 5 nM T83813 CF9VK5 24826867 Ki = 8 nM T83813 CJ7Q4O 24826868 EC50 = 10 nM T83813 CT8R9F 24826869 EC50 = 4 nM T83813 C8W9FT 24826870 EC50 = 55 nM T83813 CSDP50 24826871 EC50 = 12 nM T83813 CGQZ94 24826957 EC50 = 6 nM T83813 C5DZ6K 24826963 EC50 = 14 nM T83813 C58AMS 24829343 Ki = 358 nM T83813 CDC91N 24839550 Ki = 389.05 nM T83813 CY21RE 24841480 Ki = 940 nM T83813 CBA17N 24849050 EC50 = 23 nM T83813 CUW23K 24854106 Ki = 1500 nM T83813 CU90ZK 24861250 Ki = 2400 nM T83813 C3HK0J 24865725 Ki > 1000 nM T83813 C0O6FX 24865727 Ki > 3981.07 nM T83813 C98ZIV 24882509 IC50 = 1600 nM T83813 C0KFD3 24884789 Ki = 12.59 nM T83813 C2NT1L 24887284 Ki = 12.59 nM T83813 C2J0BI 24887285 Ki = 100 nM T83813 CB41AM 24887289 Ki = 3.981 nM T83813 CC2IJ9 24887290 Ki = 0.7943 nM T83813 CXJ90O 24887291 Ki = 7.943 nM T83813 CTDX79 24887517 Ki = 12.59 nM T83813 C6L7KS 24887518 Ki = 0.7943 nM T83813 CPY96D 24887519 Ki = 6.31 nM T83813 C90ACW 24887525 Ki = 5.012 nM T83813 CR31BN 24887527 Ki = 5.012 nM T83813 C2NVO1 24887761 Ki = 63.1 nM T83813 C17OXP 24887768 Ki = 316.23 nM T83813 C24NPA 24887966 Ki = 50.12 nM T83813 C04UDV 24887967 Ki = 5.012 nM T83813 CHA0N5 24887968 Ki = 25.12 nM T83813 CX04AI 24887970 Ki = 5.012 nM T83813 C0DX5I 24888180 Ki = 2.512 nM T83813 CO74UR 24888181 Ki = 6.31 nM T83813 CGLH34 24888182 Ki = 100 nM T83813 C6R9EH 24888183 Ki = 1.585 nM T83813 CZX93A 24888184 Ki = 0.3162 nM T83813 C1GR0V 24888185 Ki = 3.981 nM T83813 CZY2P8 24889531 Ki = 5874 nM T83813 CI53SE 24893978 Ki = 85 nM T83813 CJ63YQ 24894055 Ki = 14 nM T83813 CAOF91 24894071 IC50 = 590 nM T83813 C69AYD 24900557 Ki > 10000 nM T83813 C59FBI 24904287 Ki = 1160 nM T83813 CW4X0E 24962988 EC50 > 10000 nM T83813 C4B0FU 25070577 EC50 = 16 nM T83813 COG5H7 25070581 EC50 = 100 nM T83813 CBY3O2 25070582 EC50 = 4.5 nM T83813 CZOW25 25070907 EC50 = 125 nM T83813 C3H2FL 25070909 EC50 = 39 nM T83813 CK0FZ5 25070911 EC50 = 33 nM T83813 CO48CT 25071230 EC50 = 154 nM T83813 C9SZG1 25084025 EC50 = 14 nM T83813 C2YJX3 25099159 Ki > 10000 nM T83813 C7NJ1B 25109291 IC50 = 11700 nM T83813 CR17NY 25110703 Ki = 158.49 nM T83813 C2FY7C 25128757 Ki > 10000 nM T83813 C5NW4M 25129807 Ki > 10000 nM T83813 CQKP18 25130148 Ki = 245.47 nM T83813 CAV81B 25130157 Ki > 10000 nM T83813 C7TQ4B 25130505 Ki > 10000 nM T83813 CD04PQ 25130829 Ki > 10000 nM T83813 CM58BO 25130830 Ki = 3311.31 nM T83813 C9HYT3 25130831 Ki > 10000 nM T83813 C36NMK 25130836 Ki = 371.54 nM T83813 C1MNU0 25131483 Ki > 10000 nM T83813 CZ6NK0 25131829 Ki > 10000 nM T83813 C67QCG 25132869 Ki = 2390 nM T83813 CGBL04 25139014 Ki = 3.3 nM T83813 CJ5VX0 25140466 Ki = 62 nM T83813 CL84YJ 25141534 Ki = 86 nM T83813 CGH08V 25164128 Ki = 1995.26 nM T83813 C5C7GH 25184832 Ki = 31.62 nM T83813 C6ZY3B 25186020 Ki = 1990 nM T83813 CN06PX 25209050 Ki = 2818.38 nM T83813 CR1K8B 25209356 Ki = 1548.82 nM T83813 CLKT16 25209357 Ki > 6025.6 nM T83813 CDF83Q 25209705 Ki > 10000 nM T83813 CM2T9Y 25263297 Ki > 2000 nM T83813 CFJM71 25263302 Ki > 2000 nM T83813 C15QMB 25263320 IC50 > 1000 nM T83813 CM8TI0 26745607 IC50 = 29.4 nM T83813 C7M4DX 27545593 IC50 = 4027 nM T83813 C76LNX 27545596 IC50 = 1300 nM T83813 C1D2LR 29943048 Ki = 0.3 nM T83813 CMT4F6 30859353 IC50 = 85.8 nM T83813 CN0JB7 30859354 IC50 = 1725 nM T83813 CA93TJ 30859359 IC50 = 2071 nM T83813 C9QGK3 34257212 Ki = 74 nM T83813 CA58DL 41305446 Ki = 986 nM T83813 CG56DF 42388639 IC50 = 241 nM T83813 CH5QX6 42389467 IC50 = 4886 nM T83813 CTI9S6 42601404 EC50 = 41 nM T83813 CQR2J6 42601405 Ki = 6 nM T83813 CCYP13 42605775 Ki = 474 nM T83813 CKH3P1 42606928 Ki = 524 nM T83813 CQS4M3 42607276 Ki = 153 nM T83813 CY7W2J 42631003 Ki = 1.2 nM T83813 CV2X5B 42635027 IC50 = 57 nM T83813 CS9Q3H 42635204 IC50 = 91 nM T83813 CQ2M5S 42635387 IC50 = 215 nM T83813 CR3KM7 42635388 IC50 = 1349 nM T83813 CJ3NP5 42636941 IC50 = 72.44 nM T83813 C9QJ4Z 43386604 IC50 > 10000 nM T83813 C5ZFM0 43399328 IC50 > 10000 nM T83813 CJ41QV 44126269 Ki = 1.585 nM T83813 CQ8NV3 44214723 Ki = 2.512 nM T83813 CSVN47 44214724 Ki = 0.5012 nM T83813 CJ8F5Y 44215629 Ki = 5.1 nM T83813 CT29ZS 44216196 Ki = 1491 nM T83813 CRNL71 44225654 Ki = 13 nM T83813 C9GU8H 44250360 IC50 = 50 nM T83813 CHEX39 44250361 IC50 = 6 nM T83813 CC6G2I 44250362 IC50 = 2253 nM T83813 C2FDB1 44250364 IC50 = 1.6 nM T83813 CA8E3N 44251238 IC50 = 321 nM T83813 C3E0KJ 44251239 IC50 = 572 nM T83813 CS7G5Q 44251240 IC50 = 167 nM T83813 C15YPV 44251314 IC50 = 50 nM T83813 CV9UQ6 44251315 IC50 = 59 nM T83813 C7DH3T 44251316 IC50 = 67 nM T83813 C1ZSE5 44251317 IC50 > 10000 nM T83813 CJB10T 44251384 IC50 = 474 nM T83813 CU7Z8P 44251385 IC50 = 9441 nM T83813 C32APB 44251386 IC50 = 6369 nM T83813 C8MC0Q 44251387 IC50 = 4.5 nM T83813 C5YEA8 44251388 IC50 = 10.7 nM T83813 C0BSF6 44251389 IC50 = 1.9 nM T83813 CGAH67 44251390 IC50 = 8.2 nM T83813 CL09IQ 44263496 IC50 > 10000 nM T83813 C87MXH 44263497 IC50 > 1000 nM T83813 C83XZI 44264336 Ki = 5160 nM T83813 CIZ5W7 44267181 IC50 = 33884.42 nM T83813 C8Z1CL 44267790 IC50 = 2000 nM T83813 CIN1S4 44272400 IC50 = 660.69 nM T83813 C13QRS 44272402 IC50 = 8128.31 nM T83813 CJ15FQ 44272419 IC50 = 4168.69 nM T83813 CU35RG 44276349 Ki = 6400 nM T83813 CC2OD4 44278111 Ki > 10000 nM T83813 CRMA84 44278114 Ki > 10000 nM T83813 CF0Y4M 44278115 Ki > 10000 nM T83813 CGBY51 44287166 Ki > 10000 nM T83813 C85DJE 44287175 Ki = 42 nM T83813 C0LGX2 44287190 Ki = 300 nM T83813 C2GB5A 44287459 Ki > 10000 nM T83813 C1IWT4 44296810 IC50 = 7413.1 nM T83813 CG62JB 44298021 Ki = 125.89 nM T83813 CV5YP3 44298022 Ki = 1.585 nM T83813 CY1B3H 44298079 Ki = 100 nM T83813 CCU89I 44298080 Ki = 3.981 nM T83813 C9TS2N 44298082 Ki = 3.981 nM T83813 CY0VX7 44298086 Ki = 1 nM T83813 CSIC31 44298091 Ki = 6.3 nM T83813 CZ7BV3 44298092 Ki = 5.012 nM T83813 CO06KG 44298100 Ki = 3.162 nM T83813 C1AF0K 44298108 Ki = 2.512 nM T83813 C9AVQ8 44298118 Ki = 10 nM T83813 C6Z0QR 44298120 Ki = 1.585 nM T83813 C41MRW 44298121 Ki = 6.31 nM T83813 CP0D3F 44298126 Ki = 15.85 nM T83813 C3KUI9 44298129 Ki = 39.81 nM T83813 CH2UE9 44298138 Ki = 5.012 nM T83813 CPL7S5 44298140 Ki = 5.012 nM T83813 CJ3H6P 44298142 Ki = 3.981 nM T83813 C1SBI3 44298147 Ki = 199.53 nM T83813 CI9S7T 44298151 Ki = 31.62 nM T83813 CUQ5J7 44298157 Ki = 15.85 nM T83813 CV14AJ 44298158 Ki = 79.43 nM T83813 CG46JN 44298163 Ki = 0.5012 nM T83813 CE8C1H 44298172 Ki = 1.995 nM T83813 CS6XN2 44298173 Ki = 1 nM T83813 CO9YU5 44298175 Ki = 1.259 nM T83813 C93TDS 44298176 Ki = 1.259 nM T83813 CIP20E 44298182 Ki = 3.162 nM T83813 C5EDF3 44298186 Ki = 199.53 nM T83813 C71ZLS 44298192 Ki = 3.162 nM T83813 C0IC9T 44298193 Ki = 6.3 nM T83813 CX64BM 44298208 Ki = 1.995 nM T83813 CF1K0H 44298209 Ki = 3.162 nM T83813 C7L1FM 44298225 Ki = 1.259 nM T83813 C3NK6M 44298226 Ki = 1.585 nM T83813 CU0FL2 44298229 Ki = 0.631 nM T83813 CE1Y5J 44298230 Ki = 1.259 nM T83813 C0N3KH 44298234 Ki = 1.585 nM T83813 C9YRS1 44298236 Ki = 1.585 nM T83813 C14RQX 44298243 Ki = 1.259 nM T83813 CWC4O2 44298244 Ki = 0.7943 nM T83813 C58LBP 44298246 Ki = 5.012 nM T83813 CX2WP8 44298249 Ki = 25.12 nM T83813 C2Q5ZP 44298254 Ki = 2.512 nM T83813 CT1JY4 44299663 Ki = 125.89 nM T83813 CWS8O5 44302714 Ki = 17 nM T83813 CH65NY 44302866 Ki = 2150 nM T83813 CEF72W 44305547 IC50 = 14125.38 nM T83813 CW07BA 44306007 IC50 > 100000 nM T83813 CKY68S 44309775 Ki = 132 nM T83813 C1TKV6 44309876 Ki = 990 nM T83813 CO0X8D 44315397 Ki = 103 nM T83813 CWH8V9 44315398 Ki = 112 nM T83813 CP0C2G 44315697 Ki = 6.4 nM T83813 C7VS1O 44315715 Ki = 472 nM T83813 C6QD8K 44315716 Ki = 32 nM T83813 CNSW85 44315725 Ki = 160 nM T83813 CUJP95 44315801 Ki = 932 nM T83813 CRI0J2 44315943 Ki = 386 nM T83813 CALI20 44315965 Ki = 310 nM T83813 CW0P1Z 44315966 Ki = 223 nM T83813 CF40WU 44315993 Ki = 5.7 nM T83813 CD30XR 44315994 Ki = 43 nM T83813 COW64J 44315995 Ki = 265 nM T83813 C1GQT9 44316017 Ki = 14 nM T83813 CG5P9D 44316018 Ki = 57 nM T83813 CS25VN 44316027 Ki = 16 nM T83813 C1YCE6 44316028 Ki = 4 nM T83813 CQTB64 44316053 Ki = 793 nM T83813 CQ50LG 44316215 Ki = 4815 nM T83813 C1L3DB 44318442 IC50 > 1000 nM T83813 CV8WZ0 44318454 IC50 = 1.148 nM T83813 CMQW13 44318461 IC50 = 3.89 nM T83813 CPIT23 44318554 IC50 = 5.012 nM T83813 C75CNK 44318581 IC50 = 4.677 nM T83813 C84MTV 44318695 IC50 = 11.22 nM T83813 C8LK5W 44318820 IC50 = 6.31 nM T83813 C35OHA 44318834 IC50 = 10.23 nM T83813 CWN39R 44318841 IC50 = 30.2 nM T83813 CXJL56 44318842 IC50 = 3.02 nM T83813 C7CTF9 44318853 IC50 > 1000 nM T83813 CM39LE 44319098 IC50 = 436.52 nM T83813 C5NG8E 44319099 IC50 > 1000 nM T83813 C3RV7M 44319119 IC50 = 19.5 nM T83813 CY8L5E 44319120 IC50 = 11.75 nM T83813 CE0I4R 44319133 IC50 = 10.72 nM T83813 C9MY2X 44319134 IC50 = 7.586 nM T83813 CID52H 44321289 Ki = 111 nM T83813 CEA13Y 44323840 Ki = 39.81 nM T83813 CNYT01 44323874 Ki = 30 nM T83813 CPB89X 44323908 Ki < 10000 nM T83813 C3MXG7 44324011 Ki = 10 nM T83813 C4KGL6 44324017 Ki = 11 nM T83813 C2MSG8 44324041 Ki = 36 nM T83813 CY03UK 44324042 Ki = 8.4 nM T83813 C5IFM9 44324046 Ki = 31 nM T83813 CE3BO7 44324047 Ki = 160 nM T83813 C3C5LO 44324051 Ki = 15 nM T83813 C1NFW3 44324052 Ki = 12 nM T83813 C2W0VB 44324056 Ki = 36 nM T83813 CT48CS 44324065 Ki = 29 nM T83813 C9UR6K 44324070 Ki = 120 nM T83813 CO25PJ 44324071 Ki > 1000 nM T83813 CPZ7N8 44324079 Ki = 230 nM T83813 CF72QK 44324084 Ki = 3000 nM T83813 CM45XW 44324091 Ki = 36 nM T83813 CGOY42 44324142 Ki = 0.2512 nM T83813 CW16JD 44324737 Ki > 1000 nM T83813 CA84SN 44324765 Ki > 1000 nM T83813 COA3H4 44324800 Ki > 1000 nM T83813 CY04JW 44324972 Ki > 1000 nM T83813 C29NRF 44326124 Ki = 239 nM T83813 CHR3P2 44326125 Ki = 17 nM T83813 C0C1LX 44326219 Ki = 107.4 nM T83813 CTC70Y 44326298 Ki = 166 nM T83813 C2OZT8 44326319 Ki = 6.7 nM T83813 C8TQL9 44326320 Ki = 183 nM T83813 C0GJ3W 44326321 Ki = 31 nM T83813 CUJ74H 44326336 Ki = 24.7 nM T83813 CGE89D 44326357 Ki = 12.9 nM T83813 C3VT2B 44326358 Ki = 32.5 nM T83813 C3A1WX 44326390 Ki = 27 nM T83813 C9KA7Y 44326405 Ki = 123.5 nM T83813 CCSV14 44326407 Ki = 170 nM T83813 CY4C9X 44326422 Ki = 9.7 nM T83813 CTGR29 44326427 Ki = 677 nM T83813 CKHM97 44326433 Ki = 42.7 nM T83813 CIC4V1 44326442 Ki = 120 nM T83813 CW2A8X 44326690 Ki = 28 nM T83813 C5HW0O 44326705 Ki = 3.25 nM T83813 CN6M0P 44326751 Ki = 112.2 nM T83813 CXZL58 44326796 Ki = 416.87 nM T83813 CO3WA6 44326982 Ki = 1096.48 nM T83813 CHLE26 44327153 Ki = 354.81 nM T83813 C5M9XJ 44327167 Ki = 933.25 nM T83813 C4AI2N 44335528 Ki = 9.1 nM T83813 CV19HU 44335657 Ki = 21.4 nM T83813 CRS9N1 44335683 Ki = 10.4 nM T83813 CK4I9F 44335687 Ki = 18.3 nM T83813 CM58WP 44335695 Ki = 16.4 nM T83813 CV9G7R 44335697 Ki = 8.7 nM T83813 CKRQ49 44335713 Ki = 5.5 nM T83813 CQ3P6N 44335719 Ki = 300.1 nM T83813 CXA43J 44335732 Ki = 11.9 nM T83813 COAV62 44335766 Ki = 7.7 nM T83813 C2J0ZS 44335767 Ki = 4.9 nM T83813 C2TC7Y 44335888 Ki = 8.6 nM T83813 CPWJ26 44343212 Ki < 10000 nM T83813 C6N3XK 44345317 IC50 = 912.01 nM T83813 C2EHY6 44346844 IC50 = 2500 nM T83813 CCU89V 44350664 Ki = 1065 nM T83813 CUXH48 44352308 Ki = 2200 nM T83813 CK12OG 44359437 Ki = 229.09 nM T83813 C3LKN1 44364048 Ki = 12589.25 nM T83813 CX38YF 44364163 Ki = 1.9 nM T83813 C6M0VT 44364215 Ki = 17.8 nM T83813 C8DVZ6 44364514 Ki = 29.9 nM T83813 CMU02Q 44364616 Ki = 150 nM T83813 CJ0SZ2 44369910 Ki = 977.24 nM T83813 CZIP61 44369921 Ki = 4570.88 nM T83813 CW2X3H 44369922 Ki = 3311.31 nM T83813 CG5A2S 44369987 Ki = 141.25 nM T83813 CXIM47 44369992 Ki = 83.18 nM T83813 C1U9IX 44370125 Ki < 10000 nM T83813 CM3W6Y 44370126 Ki = 46.77 nM T83813 C2SD5H 44370139 Ki < 10000 nM T83813 CVW0F4 44377901 Ki = 639 nM T83813 C2NE7B 44377927 Ki = 90 nM T83813 C1IDK8 44377928 Ki = 417 nM T83813 CD0T3J 44377939 Ki = 259 nM T83813 CN3FA5 44377954 Ki = 222 nM T83813 C49FLN 44377965 Ki = 349 nM T83813 CZK50H 44378001 Ki = 71 nM T83813 CVH02T 44378002 Ki = 94 nM T83813 C03SDF 44378003 Ki = 53 nM T83813 C62RSW 44378016 Ki = 106 nM T83813 C6Z9UH 44378022 Ki = 501 nM T83813 C7JB3Y 44378024 Ki = 335 nM T83813 C1UY7T 44378034 Ki = 184 nM T83813 C56ZJP 44378035 Ki = 237 nM T83813 CTC75H 44378076 Ki = 320 nM T83813 C3GTV5 44378077 Ki = 82 nM T83813 CS07QF 44378128 Ki = 417 nM T83813 CWU41H 44378141 Ki = 48 nM T83813 C9R5AX 44378333 Ki = 136 nM T83813 C6EMI4 44378348 Ki = 148 nM T83813 CJF5K0 44378369 Ki = 136 nM T83813 CJ3ZM8 44378381 Ki = 106 nM T83813 C2IA3N 44383324 EC50 = 41 nM T83813 C25EZI 44383397 Ki = 33 nM T83813 C1XOB5 44387732 Ki = 49 nM T83813 CL54KN 44387733 Ki = 14 nM T83813 C80WKC 44387740 Ki = 130 nM T83813 CROA61 44387743 Ki = 844 nM T83813 C1M5OY 44387746 Ki = 49 nM T83813 CK36VZ 44387776 Ki > 4000 nM T83813 CC0WK5 44387777 Ki > 4000 nM T83813 CQ9WS8 44387780 Ki = 398 nM T83813 CQ85AW 44389003 Ki = 383 nM T83813 C4MLR3 44389645 EC50 = 3 nM T83813 CUR07Z 44389646 EC50 = 5 nM T83813 CT8Y5A 44393007 Ki = 476 nM T83813 CG9S1O 44393045 Ki = 20 nM T83813 CO6EY0 44393113 Ki = 10 nM T83813 CE03ZW 44393134 Ki = 40 nM T83813 CK85EB 44393193 Ki = 13 nM T83813 C3RV6T 44395741 Ki = 3552 nM T83813 C4B0OI 44397588 Ki = 630.96 nM T83813 C5FP0R 44397589 Ki = 1000 nM T83813 CE3G8U 44397670 Ki = 398.11 nM T83813 CQR59X 44397731 Ki = 3.8 nM T83813 C8VJ5H 44397752 Ki = 9.5 nM T83813 C8EQU9 44397832 Ki = 1.4 nM T83813 CYDA14 44397846 Ki = 2.6 nM T83813 C0FUY7 44397929 Ki = 1.5 nM T83813 CX7O9S 44401041 Ki = 4.3 nM T83813 C5XC2B 44401042 Ki = 3.7 nM T83813 CD56EA 44401105 Ki = 8.9 nM T83813 CW3PC2 44401106 Ki = 0.65 nM T83813 C9WH7P 44401164 Ki = 0.21 nM T83813 C9CWX1 44401194 Ki = 7.6 nM T83813 CXT84G 44401243 Ki = 2.4 nM T83813 CR7H0V 44401244 Ki = 17 nM T83813 CFYR54 44402349 Ki = 270 nM T83813 CFH59G 44402373 Ki = 63 nM T83813 C6J2DO 44402413 Ki = 183 nM T83813 C8FK6D 44402415 Ki > 5454 nM T83813 C9AJO5 44402449 Ki = 246 nM T83813 C9NJ8C 44402482 Ki = 4105 nM T83813 C5RX3H 44402486 Ki = 12 nM T83813 C1X3WG 44402487 Ki = 87 nM T83813 CC30BR 44402509 Ki = 183 nM T83813 C8Y7SW 44402544 Ki = 183 nM T83813 C4EAG0 44402566 Ki = 157 nM T83813 CA56WF 44402586 Ki = 41 nM T83813 C4HEJ5 44402603 Ki = 21 nM T83813 C6K3RG 44402627 Ki = 356 nM T83813 C0SCV2 44402676 Ki = 58 nM T83813 C7YPE6 44402704 Ki = 6 nM T83813 CP6DL2 44402713 Ki = 235 nM T83813 CYH87E 44402816 Ki = 72 nM T83813 C1B4QL 44403095 Ki = 267 nM T83813 C1YL7Z 44403098 Ki > 10000 nM T83813 CFV98A 44403101 Ki = 6.5 nM T83813 C6OY9S 44403102 Ki = 2833 nM T83813 CH4SX6 44403105 Ki = 1145 nM T83813 C12FIH 44403106 Ki = 9954 nM T83813 CLGA83 44403765 IC50 = 770 nM T83813 C4LKC1 44404394 Ki = 1241 nM T83813 C3EJ4G 44404396 Ki = 1077 nM T83813 CUVA58 44404608 Ki = 1258.93 nM T83813 C53KTE 44404616 Ki = 398.11 nM T83813 C4XIR6 44404619 Ki = 7.943 nM T83813 CW1BK6 44404623 Ki = 1 nM T83813 CHG15M 44404887 Ki = 73 nM T83813 CL9GC3 44404895 Ki = 468 nM T83813 CW20SO 44407327 Ki = 168 nM T83813 COY19S 44407335 Ki = 78 nM T83813 CW57QU 44407337 Ki = 86 nM T83813 C6Z5PB 44407398 Ki = 16 nM T83813 C2Q5MJ 44407440 Ki = 171 nM T83813 CR1D5Y 44407453 Ki = 39 nM T83813 CL94HP 44407460 Ki = 77 nM T83813 COH25L 44409031 Ki = 1.6 nM T83813 C4TZ7J 44409032 Ki = 52 nM T83813 C6I4CY 44409095 Ki = 104 nM T83813 CWX62Y 44409096 Ki = 2.7 nM T83813 CM6ZY0 44409097 Ki = 14 nM T83813 CJ8UB2 44409101 Ki = 16 nM T83813 C5K2ZG 44409124 Ki = 60 nM T83813 CG87PW 44409290 Ki = 3.6 nM T83813 CI69ML 44409316 Ki = 0.8 nM T83813 CMP47G 44409317 Ki = 21 nM T83813 CIPR62 44409327 Ki = 2.3 nM T83813 CPDN92 44409332 Ki = 93 nM T83813 CAO78Q 44411663 Ki = 184 nM T83813 C8NVH0 44411664 Ki = 100 nM T83813 C2Y8VK 44411667 Ki = 28 nM T83813 C38VWG 44411668 Ki = 3785 nM T83813 C5Z2IY 44411674 Ki > 4000 nM T83813 CU2EY5 44411847 Ki = 806 nM T83813 CD0OH1 44411864 Ki = 239 nM T83813 CTLN43 44411929 Ki = 449 nM T83813 CKX6D2 44411930 Ki = 404 nM T83813 CQ89KF 44411933 Ki = 2033 nM T83813 CCJ1S9 44411934 Ki = 997 nM T83813 CL28ZA 44411935 Ki = 70 nM T83813 CG13DQ 44411936 Ki = 96 nM T83813 C4MF3D 44412149 EC50 > 20000 nM T83813 CQLM69 44412150 EC50 = 180 nM T83813 C9KJV2 44412199 EC50 > 1000 nM T83813 CT3AR5 44412200 EC50 > 1000 nM T83813 CG21JM 44412308 EC50 = 519 nM T83813 C2PTL3 44412314 EC50 > 20000 nM T83813 CR5A8V 44412315 Ki > 20000 nM T83813 C0VIZ4 44412388 EC50 = 57 nM T83813 CZV87X 44412389 EC50 = 22 nM T83813 CA7CM1 44412403 EC50 = 503 nM T83813 C7R5WO 44412404 EC50 = 319 nM T83813 CA1SO2 44412405 EC50 = 420 nM T83813 CZ08EQ 44414039 Ki = 5 nM T83813 C95IMP 44414051 Ki = 199.53 nM T83813 C9W3KV 44414057 Ki = 125.89 nM T83813 C2JIS7 44414070 Ki = 125.89 nM T83813 CKM83W 44414105 Ki = 3.981 nM T83813 C34OPN 44414115 Ki = 27 nM T83813 CHC3Q5 44414116 Ki = 231 nM T83813 C3DU6O 44414117 Ki = 27 nM T83813 C8U0HV 44414118 Ki = 155 nM T83813 C1MQU7 44414127 Ki = 12.59 nM T83813 C84CDF 44414132 Ki = 12.59 nM T83813 CX10RT 44414133 Ki = 25.12 nM T83813 C6C7KD 44414136 Ki = 134 nM T83813 C5HPJ4 44414150 Ki = 100 nM T83813 CG59TD 44414151 Ki = 207 nM T83813 C9AFE0 44414154 Ki = 103 nM T83813 C6ZTK1 44414164 Ki = 7.943 nM T83813 CU29FG 44414167 Ki = 463 nM T83813 CA4MG3 44414179 Ki = 6.31 nM T83813 CT40YN 44414183 EC50 = 54 nM T83813 CWP0I4 44414184 Ki > 10000 nM T83813 CU7G6H 44414192 Ki = 7.943 nM T83813 CKTU25 44414197 Ki = 3013 nM T83813 C60DGH 44414198 Ki = 1852 nM T83813 CY41EO 44414199 Ki = 3313 nM T83813 CKU7L1 44414200 Ki = 1698 nM T83813 C5EO1B 44414209 Ki = 3.162 nM T83813 C9WJD2 44414217 Ki = 794.33 nM T83813 C6BCV8 44414218 Ki = 3381 nM T83813 C32SHA 44414219 Ki = 530 nM T83813 C10EYK 44414220 Ki = 465 nM T83813 CR3W1B 44414221 Ki = 107 nM T83813 CQ1H9S 44414233 Ki = 199.53 nM T83813 CQ13GM 44414244 Ki = 398.11 nM T83813 COY3V0 44414251 Ki = 1.259 nM T83813 CQ6K7F 44414267 Ki = 12.59 nM T83813 CT2KF0 44414290 EC50 = 11 nM T83813 C0I2TR 44414296 Ki = 155 nM T83813 CIB48J 44414297 Ki = 1141 nM T83813 CKG9P2 44414300 Ki < 1258.93 nM T83813 CF0BM8 44416391 IC50 = 10321 nM T83813 C2F3EY 44416474 IC50 = 4163 nM T83813 C70GBX 44416475 IC50 = 7467 nM T83813 C9VS6Z 44416587 IC50 = 16515 nM T83813 C4RS6H 44416627 IC50 = 14123 nM T83813 CF3HG1 44416628 IC50 = 20230 nM T83813 C8A5HU 44416629 IC50 = 4188 nM T83813 CT4DU9 44416650 IC50 > 100000 nM T83813 CGB3S0 44416689 IC50 = 14641 nM T83813 CE5MY9 44416713 IC50 = 2807 nM T83813 C0V4BK 44416737 IC50 = 3595 nM T83813 C95RCN 44416738 IC50 > 100000 nM T83813 CD9Q0Y 44416839 IC50 > 100000 nM T83813 C81JPB 44416840 IC50 > 100000 nM T83813 CPNY68 44416910 IC50 = 1313 nM T83813 CE0SK3 44416928 IC50 = 25210 nM T83813 CB9RO3 44416929 IC50 > 100000 nM T83813 CILD84 44416966 IC50 > 100000 nM T83813 CO0U5H 44417892 IC50 > 100000 nM T83813 C35KLS 44417895 IC50 > 100000 nM T83813 CA8U7N 44417896 Ki > 100000 nM T83813 CKI1W2 44417898 IC50 > 100000 nM T83813 C6UAH2 44417900 IC50 > 100000 nM T83813 CWO51Q 44417901 IC50 > 100000 nM T83813 C8GK5Q 44417904 IC50 > 100000 nM T83813 CKQ92G 44417909 Ki > 100000 nM T83813 C2XJW5 44417912 Ki > 100000 nM T83813 CPDW02 44417913 IC50 = 16000 nM T83813 C5HA7X 44417916 IC50 = 27000 nM T83813 CW1D3V 44417919 IC50 = 56000 nM T83813 C3CM4J 44417922 IC50 = 9500 nM T83813 CE96RJ 44417926 IC50 = 17000 nM T83813 CEZH78 44417928 IC50 > 100000 nM T83813 C3WT1V 44417950 Ki = 2500 nM T83813 C6F9MN 44417953 Ki = 100 nM T83813 C3P1JG 44417954 IC50 > 100000 nM T83813 C3Y5QV 44417958 IC50 > 100000 nM T83813 C3SVB8 44417960 IC50 > 100000 nM T83813 C7JFN6 44417967 Ki = 5300 nM T83813 CH6F8D 44417969 Ki = 700 nM T83813 CM2EL7 44417985 IC50 > 100000 nM T83813 CTYW15 44417987 Ki > 100000 nM T83813 C7CP8I 44417993 IC50 = 22000 nM T83813 C6Q7ZM 44418004 IC50 > 100000 nM T83813 CK9R1S 44420682 EC50 = 296 nM T83813 C6PBE9 44420683 Ki = 1450 nM T83813 C2TE3S 44425699 Ki = 10 nM T83813 CU52GB 44425701 Ki = 10 nM T83813 C9F1XP 44425702 Ki = 31.62 nM T83813 CR1QN5 44425703 Ki = 100 nM T83813 C5UZS7 44425704 Ki = 12.59 nM T83813 CN96FA 44425705 Ki = 398.11 nM T83813 C1J9MY 44425706 Ki = 79.43 nM T83813 CPI52U 44425708 Ki = 15.85 nM T83813 CNZ3M7 44425711 Ki = 125.89 nM T83813 C92AZG 44425714 Ki = 39.81 nM T83813 C7LP1B 44425717 Ki = 39.81 nM T83813 CX8TR0 44425719 Ki = 5.012 nM T83813 CJN6P4 44427818 Ki = 736 nM T83813 CW3F5H 44427820 Ki = 10.6 nM T83813 CYLO03 44427821 Ki = 96.4 nM T83813 CJY9L5 44427822 Ki = 31 nM T83813 CO46HS 44427823 Ki = 74.3 nM T83813 CFG0S3 44427824 Ki = 112 nM T83813 C7PK0M 44427825 Ki = 256 nM T83813 CDV6A3 44427826 Ki = 176 nM T83813 C65ZXC 44427827 Ki = 115 nM T83813 CZ0X7U 44427829 Ki = 2830 nM T83813 C9U8YT 44427831 Ki = 3940 nM T83813 C0C8AH 44427835 Ki = 84.3 nM T83813 C8EV3G 44427836 Ki = 25.2 nM T83813 CS9ND5 44427841 Ki = 79.3 nM T83813 COV6N3 44427842 Ki = 626 nM T83813 C7KBP0 44430566 Ki = 5.012 nM T83813 CBP57S 44430955 Ki = 251.19 nM T83813 CIZ54L 44430956 Ki = 125.89 nM T83813 C1FHD3 44430958 Ki = 199.53 nM T83813 CX0O2S 44430974 Ki = 125.89 nM T83813 CQFV73 44430976 Ki = 2.512 nM T83813 CG0CH7 44430979 Ki = 6.31 nM T83813 C14ZCW 44430984 Ki = 12.59 nM T83813 CZ3RM2 44435219 Ki = 2200 nM T83813 CKZF16 44439165 Ki < 5011.87 nM T83813 CA4HZ3 44439167 Ki = 2511.89 nM T83813 CQ18PR 44439374 Ki > 4000 nM T83813 CN9RH5 44439375 Ki > 4000 nM T83813 C2X1FS 44439377 Ki > 4000 nM T83813 CW2KQ1 44439378 Ki > 4000 nM T83813 C2J9LG 44439379 Ki = 64 nM T83813 COKH57 44439380 Ki = 220 nM T83813 CO20GU 44439381 Ki = 19 nM T83813 C4KQ8C 44439384 Ki = 1400 nM T83813 CQXS03 44439385 Ki = 160 nM T83813 C3OD9X 44441217 Ki < 10000 nM T83813 CY29KE 44441218 Ki = 109.65 nM T83813 CRPB21 44441219 Ki = 707.95 nM T83813 C6JU0E 44441222 Ki < 10000 nM T83813 CG4SU7 44441225 Ki = 741.31 nM T83813 CZL95J 44451390 Ki = 46 nM T83813 CL14SE 44451393 Ki = 20 nM T83813 C32AJU 44451422 Ki = 43 nM T83813 CT5JO6 44451429 Ki = 14 nM T83813 C3Z7FI 44451927 IC50 = 220 nM T83813 C57SBC 44451980 IC50 > 10000 nM T83813 CEST18 44451982 IC50 = 80 nM T83813 CRN4F8 44452007 IC50 = 3800 nM T83813 CG1C6X 44452142 IC50 = 1300 nM T83813 CVAU93 44452222 IC50 = 460 nM T83813 C0B3LC 44452327 IC50 = 3400 nM T83813 C63WNH 44452753 Ki = 0.51 nM T83813 CY9PG0 44452754 Ki = 0.2 nM T83813 CXCB32 44452783 Ki = 13 nM T83813 CD5J9B 44452784 Ki = 2.5 nM T83813 CI5R1U 44452785 Ki = 25 nM T83813 CX3PQ9 44452786 Ki = 59 nM T83813 C7E4KD 44452809 Ki = 4 nM T83813 CE7CQ0 44452810 Ki = 1.4 nM T83813 CNPZ39 44452831 Ki = 140 nM T83813 CSM19Y 44452832 Ki = 7.5 nM T83813 CZE3G2 44453102 Ki = 12 nM T83813 C78NHG 44453103 Ki = 300 nM T83813 C5XTC7 44453127 Ki = 20 nM T83813 C6QHC2 44453128 Ki = 5 nM T83813 CQF0U6 44453129 Ki = 2.7 nM T83813 C4L6TY 44453652 Ki = 5000 nM T83813 CVN1O4 44453877 Ki = 4000 nM T83813 CZL97F 44455426 Ki = 71 nM T83813 CYS7T4 44455943 Ki = 155 nM T83813 C6BFI0 44456033 Ki = 55 nM T83813 CG91RD 44456395 Ki = 74 nM T83813 C12XGE 44456400 Ki = 630.96 nM T83813 C5RO6E 44461290 IC50 > 1000 nM T83813 CC9JB4 44461357 IC50 = 3.802 nM T83813 CI85BO 44461456 IC50 = 13.8 nM T83813 CE12QP 44461565 IC50 = 18.62 nM T83813 CQ2IX7 44461606 IC50 = 37.15 nM T83813 C5RM2Q 44461613 IC50 = 323.59 nM T83813 CJ91XI 44461619 IC50 > 1000 nM T83813 CQX62Y 44461622 IC50 = 14.45 nM T83813 C80PVC 44461625 IC50 > 1000 nM T83813 CT09SU 44461626 IC50 > 1000 nM T83813 CR54MO 44461647 IC50 > 1000 nM T83813 C3XUF0 44461656 IC50 > 1000 nM T83813 C5P3AW 44461799 IC50 > 1000 nM T83813 C52INO 44461800 IC50 > 1000 nM T83813 C8UON6 44474625 IC50 > 1000 nM T83813 C6HVU1 44474629 IC50 > 10000 nM T83813 CJA36X 44533150 IC50 = 50 nM T83813 C3D4HR 44537940 Ki = 1070 nM T83813 CT85QK 44538690 Ki = 520 nM T83813 CJ7U3K 44554227 Ki = 1075 nM T83813 CM0I1P 44554393 Ki = 1880 nM T83813 CNHA47 44554395 Ki = 3648 nM T83813 CY18IU 44555382 Ki = 405 nM T83813 CVA67X 44568347 Ki = 3100 nM T83813 CGFE18 44572164 EC50 = 128 nM T83813 CWG32I 44572166 EC50 = 3 nM T83813 C9B3LM 44572168 EC50 = 11 nM T83813 CYS32A 44572170 EC50 = 18 nM T83813 CX93AL 44572172 EC50 = 6 nM T83813 C9PGC5 44572174 EC50 = 3.5 nM T83813 C07DQB 44572176 EC50 = 97 nM T83813 CS26GU 44572178 EC50 = 7 nM T83813 CJA7V6 44572180 EC50 = 35 nM T83813 CYOJ47 44572207 EC50 = 13 nM T83813 CV52SZ 44572252 EC50 = 301 nM T83813 CB81WN 44572254 EC50 = 1965 nM T83813 CI6U0Y 44572256 EC50 = 695 nM T83813 CX9DG3 44572258 EC50 = 1577 nM T83813 C1K5VF 44572260 EC50 > 1000 nM T83813 CO3MK4 44572262 EC50 > 1000 nM T83813 CM6HQ9 44572302 EC50 > 1000 nM T83813 C69CUA 44572304 EC50 > 1000 nM T83813 C9N4EO 44572306 EC50 = 1196 nM T83813 C0L3IQ 44572308 EC50 = 1179 nM T83813 C18IEK 44572310 EC50 > 1000 nM T83813 C34NDG 44572312 EC50 > 1000 nM T83813 C41PWR 44572314 EC50 > 1000 nM T83813 C1Y8PO 44572363 EC50 > 1000 nM T83813 CLA72W 44572365 EC50 > 1000 nM T83813 CXU7Z8 44572367 EC50 = 232 nM T83813 C6GIR9 44572369 EC50 = 136 nM T83813 CY5Q8G 44572371 EC50 = 332 nM T83813 CXJ49K 44572373 EC50 > 5000 nM T83813 CA3L9P 44572375 EC50 > 10000 nM T83813 C7WJS5 44572657 EC50 = 5.2 nM T83813 CAE0Y6 44572694 EC50 = 3416 nM T83813 CMJE86 44572696 EC50 = 5697 nM T83813 COK9N1 44572698 EC50 = 2902 nM T83813 C9QJB3 44572747 EC50 = 29 nM T83813 C6S2DJ 44572749 EC50 = 5.1 nM T83813 C97VKX 44572751 EC50 = 0.78 nM T83813 C2AQR8 44572753 EC50 = 78 nM T83813 C2RV0K 44572755 EC50 = 23 nM T83813 CKIC03 44572757 EC50 = 49 nM T83813 CQU5B9 44572759 EC50 = 26 nM T83813 CYTA39 44572761 EC50 = 161 nM T83813 C6CGB5 44572798 EC50 = 3.3 nM T83813 C20GHO 44572800 EC50 = 10 nM T83813 CJ1VI8 44572802 EC50 = 4.8 nM T83813 CLV5I8 44572804 EC50 = 30 nM T83813 C43IDZ 44572806 EC50 = 16 nM T83813 CT64CF 44572808 EC50 = 3.3 nM T83813 CU25XD 44572810 EC50 = 5.4 nM T83813 CS7KZ5 44572812 EC50 = 76 nM T83813 C6QFY7 44573002 EC50 = 138 nM T83813 CP16NR 44573004 EC50 = 135 nM T83813 C9MXB5 44573006 EC50 = 779 nM T83813 C0V1KO 44573008 EC50 = 902 nM T83813 CQ70OY 44573012 EC50 = 99 nM T83813 CE95AX 44573014 EC50 = 42 nM T83813 CEC7J9 44573016 EC50 = 87 nM T83813 CUB38Y 44573018 EC50 = 9 nM T83813 CI3V4D 44573153 Ki = 156 nM T83813 CX1N8H 44573154 Ki = 30 nM T83813 C7C5ZW 44573155 Ki = 235 nM T83813 C3L0BU 44573156 EC50 = 47 nM T83813 CD9V7Q 44573157 Ki = 1200 nM T83813 CZM8O6 44573159 EC50 = 31 nM T83813 CVSJ62 44573160 EC50 = 12 nM T83813 CF0A2J 44573161 EC50 = 28 nM T83813 C13LFI 44573162 EC50 = 14 nM T83813 CB60NZ 44573165 EC50 = 170 nM T83813 C0F5DM 44573216 Ki = 531 nM T83813 C6X3QF 44573217 Ki = 382 nM T83813 CF9X3C 44573218 Ki = 133 nM T83813 CUC43W 44573219 Ki = 10 nM T83813 C4I8AJ 44573220 Ki = 7 nM T83813 CXDU28 44573221 EC50 = 50 nM T83813 C2HS3V 44573222 Ki = 9 nM T83813 C9X6GQ 44573223 EC50 = 186 nM T83813 C7HZJ6 44573224 EC50 = 31 nM T83813 C46QXT 44573225 EC50 = 508 nM T83813 CKSA47 44573226 Ki = 15 nM T83813 CD62CX 44573227 EC50 = 273 nM T83813 CM3S4E 44573228 EC50 = 365 nM T83813 CDH04E 44573229 EC50 = 7 nM T83813 CAF64P 44573230 EC50 = 9 nM T83813 CPK71S 44573231 EC50 = 80 nM T83813 C5TKU6 44579715 Ki = 4100 nM T83813 C5NS6H 44581972 Ki = 30.2 nM T83813 CK8Z1P 44581973 Ki = 3.89 nM T83813 C3UQ9Z 44581974 Ki = 302 nM T83813 CRCH48 44582675 Ki = 53 nM T83813 CEJ4R8 44582676 Ki = 128 nM T83813 CZGP86 44582677 Ki > 10000 nM T83813 C5QB4K 44582678 Ki = 508 nM T83813 C01RCI 44582705 Ki = 497 nM T83813 CXL25V 44582706 Ki > 10000 nM T83813 C8MR1X 44582707 Ki > 10000 nM T83813 C4IT1N 44582708 Ki = 9417 nM T83813 CB0S4Z 44592109 IC50 = 29512.09 nM T83813 C43LPI 44622848 Ki = 10 nM T83813 CZHP95 44626357 EC50 = 11 nM T83813 CFOV85 45106548 IC50 = 8928 nM T83813 C0DLU3 45109862 IC50 = 599 nM T83813 CGB2Z0 45113400 Ki = 39 nM T83813 CWI23Z 45261112 Ki = 87.1 nM T83813 CJ0EF5 45261121 Ki = 125.89 nM T83813 CIQ8R1 45261133 Ki < 10000 nM T83813 C7YU6Z 45261136 Ki = 331.13 nM T83813 C2PB1G 45261140 Ki = 912.01 nM T83813 C0KXS7 45261141 Ki = 933.25 nM T83813 CDU46Z 45261169 Ki = 398.11 nM T83813 CYV2O5 45261173 Ki = 1096.48 nM T83813 C7GFY0 45261174 Ki = 363.08 nM T83813 CU6PR3 45261178 Ki = 3981.07 nM T83813 CBA1Z5 45264958 Ki = 204.17 nM T83813 CT7S9V 45264987 Ki = 81.28 nM T83813 C2J0GO 45278647 IC50 = 92 nM T83813 C7X3LG 45278648 IC50 = 344 nM T83813 CG64BP 45278720 IC50 = 160 nM T83813 CD9HF8 45278721 IC50 = 133 nM T83813 CYT87H 45278722 IC50 = 192 nM T83813 C8QK9C 45278723 IC50 = 139 nM T83813 C2M5HA 45278725 IC50 = 273 nM T83813 CXJ8L6 45278729 IC50 = 175 nM T83813 CAQ40Z 45278802 IC50 = 225 nM T83813 CARO27 45278803 IC50 = 448 nM T83813 CFG01K 45278804 IC50 = 417 nM T83813 CZ71RN 45278805 IC50 = 12 nM T83813 CFN4D9 45278806 IC50 = 66 nM T83813 CZN6M7 45278882 IC50 = 628 nM T83813 C6NT3Q 45278883 IC50 = 795 nM T83813 CA58GM 45278884 IC50 = 443 nM T83813 C21JKF 45278885 IC50 = 162 nM T83813 CS5BA4 45278886 IC50 = 466 nM T83813 C4TXE8 45278964 IC50 = 1436 nM T83813 CPI26X 45278965 IC50 = 297 nM T83813 C1NR0P 45278966 IC50 = 220 nM T83813 CYK65H 45278967 IC50 = 611 nM T83813 C0EGV6 45278968 IC50 = 638 nM T83813 CWI2S0 45279043 IC50 = 1034 nM T83813 CN7V2L 45279044 IC50 = 280 nM T83813 C2AW3R 45279045 IC50 = 615 nM T83813 CF7O1A 45279046 IC50 = 1602 nM T83813 CM46OZ 45279047 IC50 = 1298 nM T83813 CB02TI 45279127 IC50 = 342 nM T83813 CS62HT 45279130 IC50 = 21 nM T83813 CRM38P 45279134 IC50 = 149 nM T83813 CEZ53Y 45279210 IC50 = 20.9 nM T83813 CPX18C 45279212 IC50 = 61 nM T83813 CJ0X2R 45279214 IC50 = 32 nM T83813 C3NW0C 45279216 IC50 = 35 nM T83813 CX73IH 45279218 IC50 = 37 nM T83813 CGNC19 45279298 IC50 = 310 nM T83813 C8CPD7 45279300 IC50 = 63 nM T83813 CP4GI2 45279384 IC50 = 189 nM T83813 CX2ND5 45279386 IC50 = 106 nM T83813 CX5ST2 45279664 IC50 = 129 nM T83813 CKQ7S3 45279666 IC50 = 39 nM T83813 C91IRB 45279668 IC50 = 39 nM T83813 C12WRL 45279755 IC50 = 22 nM T83813 C3SUQ1 45279757 IC50 = 26 nM T83813 C63LSI 45279759 IC50 = 41 nM T83813 CT36SB 45481570 IC50 > 10000 nM T83813 CV21FS 45481572 IC50 > 10000 nM T83813 C2DKE0 45481573 IC50 > 10000 nM T83813 CS9HJ5 45481574 IC50 > 10000 nM T83813 CQI09E 45481575 IC50 = 86.9 nM T83813 CTX5P7 45481576 IC50 = 242 nM T83813 CG60OP 45481700 IC50 = 3817 nM T83813 CW6ME7 45481701 Ki = 0.89 nM T83813 C9PDX2 45481702 Ki = 2.4 nM T83813 CYK0U1 45482399 IC50 = 2052 nM T83813 C0CHF4 45482789 IC50 > 10000 nM T83813 CLO70J 45483261 Ki = 501.19 nM T83813 C7LD5K 45483269 Ki > 10000 nM T83813 CD5H2X 45483622 IC50 > 10000 nM T83813 CG8JT5 45484649 EC50 > 10000 nM T83813 CK32TH 45484650 EC50 > 10000 nM T83813 CEN01U 45484654 EC50 = 62 nM T83813 C0QP1B 45484661 EC50 = 33 nM T83813 C7JR1B 45484662 EC50 = 30 nM T83813 C2YM6L 45484673 EC50 = 31 nM T83813 C8A5GD 45484681 EC50 = 6630 nM T83813 C5MXW4 45484682 EC50 = 125 nM T83813 CG7SD9 45484686 EC50 = 48 nM T83813 CB53ZY 45484687 EC50 = 107 nM T83813 CR14VO 45484700 EC50 = 26 nM T83813 CZU53K 45484701 EC50 > 10000 nM T83813 CL16EH 45484708 EC50 > 10000 nM T83813 CIF58O 45484726 EC50 = 2930 nM T83813 CJM13Y 45484727 Ki = 2700 nM T83813 C6V3MC 45484734 EC50 = 338 nM T83813 C9K7HM 45484741 EC50 > 10000 nM T83813 CQM85L 45484742 EC50 = 176 nM T83813 CZ9A7I 45484757 EC50 > 10000 nM T83813 CNKM47 45484785 EC50 = 1020 nM T83813 CYMZ06 45484801 EC50 = 77 nM T83813 CV7OU4 45484812 EC50 > 10000 nM T83813 C32EDZ 45484826 EC50 > 10000 nM T83813 CX85DK 45484827 EC50 = 56 nM T83813 CH19MJ 45484833 EC50 = 262 nM T83813 C3HLZ6 45484841 EC50 = 899 nM T83813 CBEG69 45484848 EC50 = 163 nM T83813 C5E0BO 45484858 EC50 = 30 nM T83813 CEV19H 45484865 EC50 = 112 nM T83813 C5KV7O 45484866 EC50 = 103 nM T83813 CV9WA4 45484869 EC50 = 275 nM T83813 C5NYG0 45484870 EC50 = 73 nM T83813 CAVZ39 45484878 EC50 = 228 nM T83813 C9F3BJ 45484879 EC50 = 487 nM T83813 CCN91K 45484886 EC50 = 96 nM T83813 C8OWM9 45484888 EC50 = 493 nM T83813 CXMW65 45484896 EC50 = 319 nM T83813 C0QWC4 45484902 EC50 = 262 nM T83813 CT9WL0 45484903 EC50 = 26 nM T83813 CPR10B 45484904 EC50 > 10000 nM T83813 C2PM1O 45484908 EC50 > 10000 nM T83813 CVU0T7 45484909 EC50 = 46 nM T83813 C6BZ1Q 45484910 EC50 = 160 nM T83813 COWL37 45484927 EC50 = 361 nM T83813 C6EF4L 45484934 EC50 = 21 nM T83813 CD13VW 45484945 EC50 = 26 nM T83813 COWY41 45484946 EC50 = 64 nM T83813 CD2Z3M 45484960 EC50 > 10000 nM T83813 CG27PC 45484971 EC50 > 10000 nM T83813 CWJ51R 45484972 EC50 = 21 nM T83813 C02KME 45485697 EC50 > 9980 nM T83813 CDT1B6 45485713 EC50 > 10000 nM T83813 C80BIM 45485714 EC50 > 1920 nM T83813 C9NK6I 45485725 EC50 = 25 nM T83813 C42IXP 45485726 EC50 = 858 nM T83813 C9Q4RE 45485727 EC50 = 360 nM T83813 CLVX80 45485736 EC50 > 10000 nM T83813 CVK8W9 45485742 EC50 = 10 nM T83813 CR7Y4K 45485743 EC50 > 10000 nM T83813 CD80KX 45485751 EC50 = 164 nM T83813 CMIG41 45485752 EC50 > 10000 nM T83813 CD1YF2 45485753 EC50 > 10000 nM T83813 C2WU3I 45485754 EC50 > 2130 nM T83813 C6S3QY 45485764 EC50 = 114 nM T83813 C40MJS 45485768 EC50 > 10000 nM T83813 C0H4RN 45485769 EC50 = 510 nM T83813 CRJ8L1 45485770 EC50 > 4550 nM T83813 CNX23T 45485779 EC50 = 25 nM T83813 CFBH61 45485780 EC50 > 10000 nM T83813 CO6Z1P 45485781 EC50 = 47 nM T83813 C67AWM 45485782 EC50 > 10000 nM T83813 C2T9AC 45485786 EC50 = 407 nM T83813 CIE48J 45485787 EC50 = 101 nM T83813 C9CV1H 45486652 Ki = 403 nM T83813 CY8T1Z 45486653 Ki = 98.7 nM T83813 C1WBI2 45486654 Ki = 223 nM T83813 C3ME0C 45486656 Ki = 20 nM T83813 C2AK3J 45486657 Ki = 385 nM T83813 C0VF7N 45486658 Ki = 1230 nM T83813 CLOH56 45486664 Ki = 21.7 nM T83813 C5IV3W 45486665 Ki = 2.9 nM T83813 C0I6YB 45486671 Ki = 9 nM T83813 C12ELO 45486672 Ki = 760 nM T83813 C54GSK 45486673 Ki = 133 nM T83813 CD28FO 45486677 Ki = 213 nM T83813 C2GLK8 45486678 Ki = 102.7 nM T83813 CL6H8C 45486679 Ki = 216 nM T83813 C2TL5C 45486680 Ki = 810 nM T83813 CXQ5Z0 45486688 Ki = 3 nM T83813 CGZ62R 45486694 Ki = 9 nM T83813 C3W8EK 45486695 Ki = 8.8 nM T83813 C40DYQ 45486696 Ki = 18.9 nM T83813 CFLI93 45486697 Ki = 59.1 nM T83813 CBEF38 45486702 Ki = 21.4 nM T83813 CEF0H7 45486708 Ki = 24.3 nM T83813 CH9LW6 45486710 Ki = 66.2 nM T83813 C3LEN4 45486711 Ki = 1170 nM T83813 C7NO8W 45486713 Ki = 466 nM T83813 CI4PE6 45486714 Ki = 24 nM T83813 CXI5R2 45486715 Ki = 58.9 nM T83813 CLID23 45486716 Ki = 29.6 nM T83813 CFB39Y 45486717 Ki = 5.4 nM T83813 CT51UF 45486721 Ki = 12.7 nM T83813 CIF10P 45486722 Ki = 151 nM T83813 CUZ79F 45486723 Ki = 187 nM T83813 CA39DM 45486724 Ki = 50.7 nM T83813 C9X2NP 45486725 Ki = 98 nM T83813 C3LX5I 45486726 Ki = 210 nM T83813 CTC15H 45486727 Ki = 147 nM T83813 CR25SJ 45486729 Ki = 481 nM T83813 CES7G9 45486731 Ki = 104 nM T83813 CX74NQ 45486732 Ki = 53.2 nM T83813 C4RTL1 45486733 Ki = 37.8 nM T83813 CM08SQ 45486737 Ki = 1090 nM T83813 CFEK40 45486738 Ki = 11 nM T83813 CIV92F 46214153 Ki = 760 nM T83813 C5FQ4S 46224879 Ki = 0.4786 nM T83813 CY82LR 46227396 IC50 = 1396 nM T83813 C6YE4Q 46228417 IC50 = 710 nM T83813 C2Z6MJ 46228421 IC50 > 500 nM T83813 CF6BQ7 46228422 Ki = 20 nM T83813 CQX71P 46228423 Ki = 4 nM T83813 C4UN8O 46228425 Ki = 0.6 nM T83813 C9Q5AP 46228429 IC50 = 126 nM T83813 C23DJK 46228430 Ki = 10 nM T83813 CG82KB 46228432 IC50 = 540 nM T83813 C8TJK9 46228434 Ki = 1 nM T83813 CTES15 46228437 Ki = 1.5 nM T83813 CZ5MW9 46228438 EC50 = 0.1 nM T83813 CZ4DR0 46228439 Ki = 3 nM T83813 CI7KO8 46228440 IC50 = 410 nM T83813 CO9AK2 46228442 Ki = 28 nM T83813 C98NCA 46230046 EC50 = 137 nM T83813 C3LMQ6 46230047 EC50 = 133 nM T83813 C0D4IZ 46230048 EC50 = 4197 nM T83813 C6UMX7 46230049 EC50 = 43 nM T83813 C87JZL 46230094 EC50 = 110 nM T83813 CINK61 46230095 EC50 = 92 nM T83813 C6N7AF 46230096 EC50 > 10000 nM T83813 C7WO5P 46230097 EC50 = 16 nM T83813 CP0T5Y 46230098 EC50 = 2 nM T83813 CPA62G 46230099 EC50 = 1.8 nM T83813 CWQD49 46230100 Ki = 6.5 nM T83813 CXUL12 46232559 IC50 = 50.7 nM T83813 CU2RG8 46232560 IC50 = 156.2 nM T83813 C9RQ8U 46232586 IC50 = 293.6 nM T83813 C2B3ZP 46232587 IC50 = 45.7 nM T83813 C3I8TO 46232588 IC50 = 79 nM T83813 COW9V6 46232589 IC50 = 200 nM T83813 CGV2J5 46232620 IC50 = 33 nM T83813 CWHG97 46232621 IC50 = 40 nM T83813 CUQW08 46232622 IC50 = 65 nM T83813 C5REP7 46232623 IC50 = 70 nM T83813 C2QOW0 46232652 IC50 = 66 nM T83813 C9I7XS 46232653 IC50 = 24 nM T83813 C5D0BH 46232654 IC50 = 842.7 nM T83813 C5PAL9 46232689 IC50 = 117.9 nM T83813 CT5C0M 46232690 IC50 = 38.8 nM T83813 CF53BL 46232691 IC50 = 135.8 nM T83813 CE1ID7 46232729 IC50 = 66.5 nM T83813 CN0CO9 46232730 IC50 = 1459 nM T83813 C0VXA5 46232731 IC50 = 565 nM T83813 C1C4OF 46232732 IC50 = 1981 nM T83813 CMR8O9 46232770 IC50 = 1943 nM T83813 CTY9H7 46232771 IC50 = 691 nM T83813 C5TBE8 46232772 IC50 = 1976 nM T83813 COH03R 46232773 IC50 = 1034 nM T83813 CZ2W7X 46232817 IC50 = 723 nM T83813 C0N4YP 46232818 IC50 = 479 nM T83813 CTJ89I 46232819 IC50 = 549 nM T83813 CS98DM 46232820 IC50 = 304 nM T83813 C8P3HD 46232858 IC50 = 343 nM T83813 CP04TS 46232859 IC50 = 2159 nM T83813 C8W0IJ 46232860 IC50 = 8312 nM T83813 CF5M2T 46232861 IC50 = 694 nM T83813 C21CHG 46232975 IC50 = 4755 nM T83813 CO41KX 46232976 IC50 = 200 nM T83813 CIK94R 46232977 IC50 = 539 nM T83813 CB67ST 46232978 IC50 = 942 nM T83813 CRU0F7 46233014 IC50 = 90 nM T83813 C42SVX 46700866 IC50 = 8800 nM T83813 CD0K6E 46700867 IC50 = 4500 nM T83813 C6K0MF 46830177 Ki = 0.9 nM T83813 C5TC2S 46830335 IC50 > 10000 nM T83813 C1K7FL 46830336 IC50 > 10000 nM T83813 C7G3AC 46833072 Ki = 9250 nM T83813 CICY27 46833073 Ki > 10000 nM T83813 CBO0R4 46833074 Ki = 3380 nM T83813 C6G1DY 46833075 Ki > 10000 nM T83813 CW6O7R 46833076 Ki > 10000 nM T83813 CI4DB9 46833077 Ki > 10000 nM T83813 CWU46E 46833370 Ki > 10000 nM T83813 CZY08H 46833371 Ki = 5614 nM T83813 CRCS34 46833372 Ki = 8600 nM T83813 C5L9IJ 46833373 Ki = 5890 nM T83813 CXIE19 46833374 Ki > 10000 nM T83813 C8WCT0 46833678 Ki = 2347 nM T83813 C1N4KX 46842383 IC50 > 10000 nM T83813 CC62SX 46866711 IC50 = 100 nM T83813 CHIW05 46880277 IC50 = 156 nM T83813 CK8A1O 46880462 Ki > 10000 nM T83813 C9KDP4 46880463 Ki > 10000 nM T83813 CODR73 46880498 Ki > 10000 nM T83813 CHJ5Y6 46880566 Ki > 10000 nM T83813 CE9PG2 46880567 Ki > 10000 nM T83813 C01PGO 46880568 Ki > 10000 nM T83813 CS7L4X 46880569 Ki > 10000 nM T83813 C0PXY7 46880628 Ki > 10000 nM T83813 CD37LU 46880629 Ki > 10000 nM T83813 CUY89F 46880630 Ki > 10000 nM T83813 C4P6XS 46880631 Ki > 10000 nM T83813 CJ53KF 46880672 Ki > 10000 nM T83813 CYJC08 46880673 Ki > 10000 nM T83813 C1RI9O 46880674 Ki > 10000 nM T83813 CI96SR 46884034 Ki = 4 nM T83813 C2C7OU 46884035 Ki = 83 nM T83813 C6EL4F 46884036 Ki = 324 nM T83813 CW0SU5 46884037 Ki = 643 nM T83813 C5U2EC 46884038 Ki = 585 nM T83813 CEUD30 46884098 Ki = 4.4 nM T83813 CF2TL4 46884099 Ki = 8 nM T83813 CNET68 46884100 Ki = 23 nM T83813 C8Y0IG 46884101 Ki = 20 nM T83813 C5BFY9 46884102 EC50 = 1 nM T83813 C1ORQ0 46884137 Ki = 25 nM T83813 C3BW2P 46884138 Ki = 1.7 nM T83813 CB8GE1 46884818 IC50 > 10000 nM T83813 C4MQ0A 46884856 IC50 > 10000 nM T83813 CCNT25 46884898 IC50 > 10000 nM T83813 C3MSG2 46885027 IC50 > 10000 nM T83813 CB7XI0 46885213 IC50 > 10000 nM T83813 C3MPJ7 46890808 Ki = 184 nM T83813 C60OHX 46901596 Ki > 10000 nM T83813 C4VIO7 46901598 Ki > 10000 nM T83813 CT5S4Q 46901603 Ki > 10000 nM T83813 C7KO6F 46901762 Ki > 10000 nM T83813 CYQ3L9 46901908 Ki = 3866 nM T83813 CX3AE0 46901909 Ki = 3714 nM T83813 C2ULG1 46927928 IC50 = 64 nM T83813 CK21VU 46927929 IC50 = 86.15 nM T83813 CG7WR2 46933089 Ki = 50.12 nM T83813 CW4N5K 46933090 Ki = 125.89 nM T83813 CZO5F8 46933091 Ki = 501.19 nM T83813 CH86DQ 46933237 Ki = 41 nM T83813 CX7R3H 46933845 EC50 = 0.7244 nM T83813 CUTX67 46934428 IC50 = 4 nM T83813 CV8A5L 46937339 EC50 = 21 nM T83813 CPFY62 49782791 Ki = 3.1 nM T83813 CKGU71 49782792 Ki = 26 nM T83813 CNE84I 49782794 Ki = 8 nM T83813 CS09QO 49782998 Ki = 93 nM T83813 C2LZJ0 49783209 Ki = 685 nM T83813 C57SMG 49783415 Ki > 10000 nM T83813 C0TG6I 49783419 Ki = 8363 nM T83813 CD53RT 49833882 Ki > 1995.26 nM T83813 C5Y4DE 49833883 Ki = 63.1 nM T83813 CGT73Y 49833884 Ki = 31.62 nM T83813 CKL16R 49833886 Ki = 501.19 nM T83813 C3KSZ8 49834050 Ki > 794.33 nM T83813 C9QS2K 49834051 Ki > 794.33 nM T83813 CF4SX0 49834052 Ki = 501.19 nM T83813 C52GPW 49834053 Ki = 316.23 nM T83813 CO20JE 49836187 Ki > 1995.26 nM T83813 CG0LF8 49836189 Ki > 1995.26 nM T83813 C0UI3V 49836294 Ki = 158.49 nM T83813 CT7CV0 49836295 Ki = 158.49 nM T83813 CVG9X5 49836296 Ki = 316.23 nM T83813 C5E2ZK 49836298 Ki = 199.53 nM T83813 CYJW87 49836299 Ki = 63.1 nM T83813 C0MS8L 49836300 Ki = 15.85 nM T83813 CR40BA 49836386 IC50 > 10000 nM T83813 CKS86Q 49836409 Ki = 125.89 nM T83813 C8E6WA 49836410 Ki = 1000 nM T83813 CE0PN6 49836411 Ki > 2511.89 nM T83813 C0I4EC 49836412 Ki = 31.62 nM T83813 C5HU1D 49836413 Ki = 1584.89 nM T83813 C1UGC7 49836414 Ki = 316.23 nM T83813 C5ZV2Y 49836522 Ki = 199.53 nM T83813 C1JTH9 49836524 Ki = 15.85 nM T83813 C90XTY 49836525 Ki = 19.95 nM T83813 CK5QW9 49836526 Ki = 19.95 nM T83813 C8RL7C 49836527 Ki > 1995.26 nM T83813 CNM9X8 49836528 Ki = 63.1 nM T83813 COK75S 49836633 Ki = 6.31 nM T83813 CZ6F7L 49836634 Ki > 1995.26 nM T83813 CRM28S 49836635 Ki = 251.19 nM T83813 CA6QB8 49836636 Ki > 1995.26 nM T83813 CB81YG 49836637 Ki = 1000 nM T83813 CEBP01 49836737 Ki > 1995.26 nM T83813 CY1UR9 49836739 Ki > 1995.26 nM T83813 C26NFU 49836741 Ki > 1995.26 nM T83813 C4R2YS 49850567 Ki > 1584.89 nM T83813 C07JTU 49850570 Ki = 794.33 nM T83813 CK68QR 49850672 Ki = 794.33 nM T83813 CN5XR1 49850772 Ki = 1995.26 nM T83813 CR4EZ0 49850870 Ki = 3162.28 nM T83813 C5K4EC 49850872 Ki = 1000 nM T83813 C8AW0R 49850874 Ki = 794.33 nM T83813 CIA24C 49863566 IC50 = 1392 nM T83813 CZB85K 49863567 IC50 = 1021 nM T83813 C7V6WO 49863654 IC50 = 349 nM T83813 CH36GC 49863692 IC50 = 633 nM T83813 C39VLG 49863693 IC50 = 782 nM T83813 CKF87D 49863694 IC50 = 493 nM T83813 CZF5Q2 49863695 IC50 = 233 nM T83813 CFTZ59 49863717 IC50 = 653 nM T83813 C7IK0Y 49863741 IC50 = 324 nM T83813 C1GR9V 49863742 IC50 = 633 nM T83813 CRQ7U4 49863743 IC50 = 1408 nM T83813 CF2TO6 49863774 IC50 = 452 nM T83813 C7Y8OQ 49863775 IC50 = 977 nM T83813 C24EAI 49863776 IC50 = 1006 nM T83813 CM72WN 49863778 IC50 = 619 nM T83813 CZR6T8 49863794 IC50 = 420 nM T83813 CB13XF 49863795 IC50 = 12 nM T83813 C6GB5R 49863847 IC50 = 13 nM T83813 C8PQB0 49863849 IC50 = 16 nM T83813 C1EKY3 49863851 IC50 = 75 nM T83813 CS80EL 49863853 IC50 = 16 nM T83813 C4HB5K 49863957 IC50 = 420 nM T83813 C18ICN 49863958 IC50 = 2227 nM T83813 C8H6GV 49863959 IC50 = 1145 nM T83813 CMRQ30 49863961 IC50 = 109 nM T83813 C9KIU1 49864289 IC50 = 6 nM T83813 CCS5D6 49864290 IC50 = 11 nM T83813 CS9L4X 49864291 IC50 = 168 nM T83813 CHO9C0 49864292 IC50 = 32 nM T83813 C6E2DI 49864314 IC50 = 34 nM T83813 CU0TJ6 49864530 IC50 = 4638 nM T83813 C9FD2E 49864599 IC50 = 1715 nM T83813 CVY4O3 49864600 IC50 > 10000 nM T83813 CJF6T5 49864601 IC50 = 467 nM T83813 C90MTG 49864602 IC50 = 21 nM T83813 CK7IY8 49864663 IC50 = 4164 nM T83813 CWC3N4 49864664 IC50 > 10000 nM T83813 CPVM78 49864665 IC50 = 97 nM T83813 CSQ4O5 49864666 IC50 > 10000 nM T83813 C2VW8O 49864686 IC50 = 106 nM T83813 CWA07N 49864687 IC50 = 243 nM T83813 C5U9XC 49864688 IC50 = 420 nM T83813 CFLE15 49864689 IC50 = 462 nM T83813 CLD20Y 49864690 IC50 = 7702 nM T83813 C5R1BM 49864721 IC50 = 159 nM T83813 C5BCS4 49864722 IC50 = 36 nM T83813 CKZO79 49864723 IC50 = 7 nM T83813 C74LZS 49864724 IC50 = 16 nM T83813 CZ2SA8 49864841 Ki = 19.95 nM T83813 C2OCZ3 49864885 Ki > 1995.26 nM T83813 CS4Z8A 49864886 Ki = 158.49 nM T83813 CN8XT2 49865829 Ki = 5171 nM T83813 C1FMH5 49865830 Ki > 10000 nM T83813 C1CX5F 49865831 Ki > 10000 nM T83813 C8RYW1 49865832 Ki > 10000 nM T83813 C5ED3T 49865833 Ki > 10000 nM T83813 CAU15V 49865885 Ki > 10000 nM T83813 CLS0F3 49865886 Ki > 10000 nM T83813 CIG69Z 49865887 Ki > 10000 nM T83813 C5YEG8 49865888 Ki > 10000 nM T83813 CXP91V 49865889 Ki > 10000 nM T83813 C98TVK 49865890 Ki > 10000 nM T83813 C2RY0J 50878551 EC50 = 9.333 nM T83813 C1W6TV 50898777 Ki > 10000 nM T83813 CXMZ73 50898778 Ki > 10000 nM T83813 CYGD56 50899654 IC50 = 610 nM T83813 CBLK68 50899745 IC50 = 227 nM T83813 CJI9U2 50899747 IC50 = 81 nM T83813 CU7TK4 50899749 IC50 = 148 nM T83813 CW9SV5 50942111 EC50 = 95 nM T83813 CX48AD 51002362 Ki = 2243 nM T83813 C8TA1J 51003550 IC50 = 558 nM T83813 CQ1UJ7 51003551 IC50 = 30 nM T83813 CGMI37 51003586 IC50 = 4 nM T83813 CE4KP1 51050257 Ki > 10000 nM T83813 CI90RZ 51094588 EC50 > 10000 nM T83813 C2HGK8 51122451 Ki > 1000 nM T83813 CX5ZB8 52940714 IC50 = 1266 nM T83813 CE26GV 52941856 IC50 = 575 nM T83813 CH86KJ 52941866 IC50 = 1178 nM T83813 C7OZN4 52944115 Ki = 7.943 nM T83813 CZ21PJ 52944292 IC50 = 135 nM T83813 C2TK7W 52945494 IC50 = 1548 nM T83813 CPD0Y9 52945500 IC50 = 1170 nM T83813 CL7OG0 52945537 IC50 = 2688 nM T83813 CHFI03 52945539 IC50 = 494 nM T83813 CNQF49 52945978 Ki = 100 nM T83813 CRH43M 52946023 Ki = 11 nM T83813 CRH1P6 52947969 IC50 = 30 nM T83813 CFN80U 52949206 IC50 = 2049 nM T83813 CW2LS0 53303985 Ki = 239.88 nM T83813 C0AY5O 53317923 EC50 = 65 nM T83813 CC0T6E 53317924 EC50 = 188 nM T83813 C1T3AI 53317925 EC50 = 8.4 nM T83813 C61DNP 53320009 IC50 = 5187 nM T83813 C9ZDR5 53320010 IC50 = 438 nM T83813 C3CT4H 53320653 EC50 = 362 nM T83813 C40VGZ 53321865 EC50 = 37 nM T83813 C7LE3I 53321947 EC50 = 764 nM T83813 CC3DB8 53321948 EC50 = 25 nM T83813 CQLK01 53322638 IC50 = 19 nM T83813 CUNP37 53323196 EC50 = 211 nM T83813 C32YWL 53324045 Ki = 2131 nM T83813 CJ9I7U 53324165 EC50 = 63 nM T83813 CQVR02 53324327 EC50 = 574 nM T83813 CN8X4Z 53324629 EC50 = 4564 nM T83813 C8DL1N 53324630 EC50 = 5 nM T83813 CRQF15 53325242 Ki = 1712 nM T83813 C2ZFP8 53325935 EC50 = 5.4 nM T83813 CNE6Q8 53325936 EC50 = 18 nM T83813 C8VUJ6 53325937 EC50 = 23 nM T83813 CMB09H 53325938 EC50 = 84 nM T83813 C3MEG7 53327952 Ki = 280 nM T83813 CZL9W7 53327953 Ki = 776.25 nM T83813 CCL48Y 53327973 Ki = 467.74 nM T83813 CT5MJ8 53327974 Ki = 457.09 nM T83813 C73SCE 53327975 Ki = 346.74 nM T83813 C5J8IG 53327976 Ki = 1096.48 nM T83813 C73THY 53327977 Ki = 457.09 nM T83813 CGV7O2 53327979 Ki = 1200 nM T83813 C4G7RQ 53327999 Ki = 870 nM T83813 CU9ON5 53328000 Ki = 370 nM T83813 C1HU7Y 53328001 Ki = 2884.03 nM T83813 CG24AT 53381002 Ki > 10000 nM T83813 CY18NZ 54189746 IC50 = 4260 nM T83813 C48CEL 54576149 IC50 = 546.4 nM T83813 C6PDR1 54576153 IC50 = 425 nM T83813 CX4OJ6 54576369 IC50 = 609 nM T83813 CA0O2M 54576371 IC50 = 1184 nM T83813 CY67DI 54576594 IC50 > 10000 nM T83813 CWUK35 54576597 IC50 = 653.7 nM T83813 C40IGO 54576800 IC50 = 170 nM T83813 CP4CV6 54576803 IC50 = 1001 nM T83813 C4H3DT 54576804 IC50 = 184.6 nM T83813 CG24OE 54577010 IC50 = 286 nM T83813 CYZX34 54577012 IC50 = 290 nM T83813 C2WQE9 54577014 IC50 = 103 nM T83813 C83FGA 54577018 IC50 = 10140 nM T83813 CWA58G 54577234 IC50 = 193.4 nM T83813 CA83GC 54577236 IC50 = 116 nM T83813 CJA0P6 54577243 IC50 = 609.6 nM T83813 C0NBJ7 54577435 IC50 = 146 nM T83813 CYW50O 54577439 IC50 = 283 nM T83813 C8YAZ5 54577443 IC50 = 190.9 nM T83813 C3P0LZ 54577446 IC50 = 593 nM T83813 CA94CQ 54577447 IC50 = 227 nM T83813 CE64WZ 54577448 IC50 = 1779 nM T83813 CJS4H9 54577449 IC50 = 193 nM T83813 CMR6C3 54577665 IC50 = 130 nM T83813 CS9G8L 54577668 IC50 = 96 nM T83813 CA8J7E 54577670 IC50 = 1031 nM T83813 C3P2KF 54577879 IC50 = 104 nM T83813 C9GFP0 54577882 IC50 = 124 nM T83813 C6KY9M 54577886 IC50 = 323.7 nM T83813 CES29I 54578098 IC50 = 68 nM T83813 CQ67LT 54578099 IC50 = 238 nM T83813 CAPC31 54578102 IC50 = 64.1 nM T83813 C12XBJ 54578547 IC50 = 159 nM T83813 CP24ZC 54579002 IC50 = 3996 nM T83813 CXQK40 54579004 IC50 = 237 nM T83813 CZC81X 54579005 IC50 = 68 nM T83813 CSW18T 54579229 IC50 = 2741 nM T83813 C5HC0P 54579233 IC50 = 525 nM T83813 CA4E9U 54579450 IC50 > 10000 nM T83813 C3L1IB 54579451 IC50 = 595.4 nM T83813 C9JZ7K 54580137 Ki = 180 nM T83813 C6WR0E 54580776 Ki = 1850 nM T83813 CSK36H 54581122 Ki = 280 nM T83813 C74EGT 54581791 EC50 = 192 nM T83813 CWB48T 54582158 Ki = 68 nM T83813 C5VS4M 54582159 Ki = 61 nM T83813 C8QLJ2 54583109 Ki = 77 nM T83813 C3GCR2 54583742 EC50 = 194 nM T83813 CV1IF6 54583743 Ki = 84 nM T83813 CT49MZ 54584107 Ki = 74 nM T83813 CU2VZ8 54584108 Ki = 49 nM T83813 CVYS68 54584720 EC50 = 110 nM T83813 CIC92Q 54584721 EC50 = 310 nM T83813 CCN6S2 54585045 Ki = 57 nM T83813 CUCO10 54585651 EC50 = 1900 nM T83813 C9DP2X 54585652 EC50 = 380 nM T83813 C46WCJ 54585653 EC50 = 300 nM T83813 C2SDF5 54586019 Ki = 120 nM T83813 COJ5R8 54586020 Ki = 83 nM T83813 CZE6V0 54586996 Ki = 91 nM T83813 C4VA8X 54586997 Ki = 49 nM T83813 C96UOS 54587668 Ki = 305 nM T83813 CTE1V3 54587669 EC50 = 210 nM T83813 CW89BT 56595402 Ki > 1000 nM T83813 C4C3XQ 56595529 Ki > 1000 nM T83813 CA54LD 56597090 Ki = 0.6 nM T83813 CH37LU 56663451 IC50 > 10000 nM T83813 CUMB38 56834972 IC50 = 55 nM T83813 CB0P9N 56944383 Ki = 540 nM T83813 CHN2F6 56949640 Ki > 10000 nM T83813 C1TC7Q 56963799 Ki > 10000 nM T83813 C6H9UV 57345617 Ki = 2434 nM T83813 CZU6L2 57345618 Ki > 10000 nM T83813 CK9G8H 57345619 Ki = 4097 nM T83813 C91XDJ 57381548 Ki = 1000 nM T83813 COR06S 57381549 Ki = 144 nM T83813 C6S0IE 57390695 Ki = 5920 nM T83813 COA60R 57391358 Ki = 496 nM T83813 C7UC1O 57391359 Ki = 997 nM T83813 CNLK91 57391360 Ki = 391 nM T83813 CV7N9Z 57391692 IC50 = 5733 nM T83813 CQO80V 57391693 IC50 = 579 nM T83813 CTX71S 57393122 Ki = 1360 nM T83813 CTF5M7 57393393 IC50 > 10000 nM T83813 C9QT8H 57393432 IC50 = 164 nM T83813 CADH19 57394285 Ki = 2529 nM T83813 CKL2B3 57394858 Ki = 467 nM T83813 CNGJ92 57394859 Ki = 394 nM T83813 CM7FS9 57394860 Ki = 739 nM T83813 CVZ5Q2 57395160 IC50 = 603 nM T83813 CY4JR5 57396622 Ki = 152 nM T83813 C6HBG0 57396813 Ki = 19000 nM T83813 C80SUY 57396884 IC50 = 1940 nM T83813 C5FU4X 57396934 IC50 > 10000 nM T83813 CQ0D5K 57398388 Ki = 246 nM T83813 CNZ6E8 57398389 Ki = 2877 nM T83813 CM8S6E 57398674 IC50 = 523 nM T83813 CBXQ64 57398675 IC50 = 1820 nM T83813 CJ41PW 57399432 Ki = 1420 nM T83813 CO3B4P 57399494 Ki = 3775 nM T83813 C0R6QM 57400053 Ki = 194 nM T83813 CN7G6D 57400054 Ki = 717 nM T83813 CO98FL 57400055 Ki = 581 nM T83813 CUQZ68 57400351 IC50 = 2422 nM T83813 CHG0A7 57401861 Ki = 575 nM T83813 CA51WJ 57401862 Ki = 596 nM T83813 C3SB2U 57401863 Ki = 6900 nM T83813 CE5QB7 57403569 Ki = 910 nM T83813 C68VZL 57403570 Ki = 190 nM T83813 CLV07S 57403571 Ki = 682 nM T83813 CSWR29 57403903 IC50 = 1195 nM T83813 CWBG94 57403981 Ki = 4623 nM T83813 CQB6F9 57456630 Ki > 1000 nM T83813 CDG58R 57799306 EC50 = 2.6 nM T83813 CS6BM2 57799321 EC50 = 62 nM T83813 CUYA69 57799324 EC50 = 2.2 nM T83813 CYPG17 57799326 EC50 = 27 nM T83813 C0M5PN 57873490 Ki > 1000 nM T83813 CH1BN8 57873491 Ki = 73.4 nM T83813 CI5UO1 57873492 Ki = 602 nM T83813 C2D9HA 57873499 Ki > 1000 nM T83813 C81MLX 57873504 Ki > 1000 nM T83813 C7L9IE 57873508 Ki = 57 nM T83813 CZRL39 57873513 Ki = 479 nM T83813 C98WTS 57873515 Ki = 61 nM T83813 C6BHT3 57873518 Ki = 475 nM T83813 CPX17D 57873520 Ki = 6 nM T83813 C54ROE 57873522 Ki > 1000 nM T83813 CM7PI1 57873525 Ki > 1000 nM T83813 CMUR21 57873527 Ki = 450 nM T83813 CO5Y9Q 57873531 Ki = 17 nM T83813 CHB3D6 58405078 Ki = 1109 nM T83813 CX2HU7 58405183 Ki = 38 nM T83813 C3TGM7 58911532 Ki = 77 nM T83813 CFC79Z 58911534 EC50 = 28 nM T83813 CD8JI3 58911579 EC50 = 64 nM T83813 CR19FG 58911582 EC50 = 12 nM T83813 C4Z5UB 58911604 EC50 = 171 nM T83813 C49INW 58911644 EC50 = 320 nM T83813 CPC3Z0 58911653 EC50 = 92 nM T83813 CNEQ36 58911666 EC50 = 33 nM T83813 CJTR58 58911668 EC50 = 48 nM T83813 CG52WR 58911681 EC50 = 1744 nM T83813 C2KP7G 59012632 EC50 = 168 nM T83813 CRKS62 59312249 EC50 = 112 nM T83813 CO6P7J 59312265 EC50 > 10000 nM T83813 C31HCO 59312310 EC50 = 51 nM T83813 CB9GC6 60165412 Ki = 2140 nM T83813 CI5PM3 60165413 Ki = 3738 nM T83813 C2Q5VD 60165416 Ki = 6210 nM T83813 C9JL3F 60165418 Ki > 10000 nM T83813 C31PEN 60165535 Ki = 6265 nM T83813 C5RUP6 60167166 Ki = 4647 nM T83813 CY8QF1 60167503 IC50 = 10000 nM T83813 CI30FT 60204111 Ki = 311 nM T83813 CWSA08 60204112 Ki > 1000 nM T83813 CC3Y9Z 67097734 EC50 > 10000 nM T83813 C6M0ZO 67098465 EC50 > 10000 nM T83813 C1LEH8 67268994 Ki = 799 nM T83813 CI8SB4 67320583 IC50 = 5257 nM T83813 C6V0RG 68690817 EC50 = 600 nM T83813 C1R7EY 68691189 EC50 = 610 nM T83813 CZFT98 68803474 EC50 = 251.19 nM T83813 C5FAB3 69314950 Ki = 15.9 nM T83813 CKM14W 69432471 Ki = 83 nM T83813 CHKP64 69433076 Ki = 110 nM T83813 C5P0ME 69471377 Ki = 532 nM T83813 C4FZ6G 69514548 Ki = 150 nM T83813 CFND58 69588506 Ki = 507 nM T83813 CI16QU 69616387 Ki = 179 nM T83813 C7FMA4 70676458 Ki = 2920 nM T83813 CQFW61 70681340 EC50 = 7240 nM T83813 CTA37Q 70681342 EC50 = 254 nM T83813 C56LVZ 70681346 EC50 = 1210 nM T83813 CB62XQ 70683433 EC50 = 18 nM T83813 CH29OT 70685538 EC50 = 8710 nM T83813 C3JVF5 70685540 EC50 = 978 nM T83813 C6FY2A 70687202 Ki = 13 nM T83813 C7QUO3 70687695 EC50 = 24 nM T83813 CE6M1I 70688018 IC50 = 3.1 nM T83813 C5PT8Y 70689809 EC50 = 3800 nM T83813 C20MDO 70689811 EC50 = 3470 nM T83813 CH40WS 70691529 EC50 = 163 nM T83813 CYN75R 70693926 EC50 = 55 nM T83813 CZC8S7 70693928 EC50 = 304 nM T83813 C9P7YD 70695555 Ki = 180 nM T83813 CVU08A 70695812 Ki = 1850 nM T83813 C51JUA 70696049 EC50 = 3310 nM T83813 C6FY7N 70696051 EC50 = 2190 nM T83813 CW71LQ 70696356 IC50 = 120 nM T83813 CYAS63 70697549 EC50 = 4.677 nM T83813 CC43QK 71151588 Ki > 1000 nM T83813 CM6EL0 71449808 IC50 = 120 nM T83813 C3XNC2 71450247 Ki = 729 nM T83813 C9VZ8J 71450550 Ki = 835 nM T83813 CKF1J3 71451614 IC50 > 40000 nM T83813 C1S6JD 71451615 IC50 = 1250 nM T83813 CKXC07 71451616 IC50 = 600 nM T83813 C4TWS5 71452172 Ki > 10000 nM T83813 C7W5XO 71455160 IC50 > 40000 nM T83813 CAQF34 71455625 Ki = 492 nM T83813 C7MNB5 71457264 Ki = 3124 nM T83813 CMJ1O9 71457409 Ki = 341 nM T83813 C1EA6Q 71458069 Ki = 400 nM T83813 C28MWU 71458824 IC50 = 10 nM T83813 CH9G5O 71458826 IC50 = 390 nM T83813 CS83IF 71459269 Ki = 400 nM T83813 CK5T4P 71459604 Ki = 1404 nM T83813 CG0WO9 71459954 Ki = 235 nM T83813 C63YLA 71461049 Ki > 10000 nM T83813 CJD96I 71461050 Ki = 1049 nM T83813 C5B2WL 71461603 Ki = 2.2 nM T83813 C0AD3M 71462344 IC50 = 180 nM T83813 C4P3JU 71462776 Ki = 772 nM T83813 C3GUQ2 71462777 Ki = 2793 nM T83813 CKX5O8 71463061 Ki = 4480 nM T83813 CHY78V 71562549 EC50 > 1000000 nM T83813 CR8Q1X 71562552 EC50 > 1000000 nM T83813 CF4XJ2 71562661 EC50 = 100 nM T83813 C29VZI 71562662 Ki > 300000 nM T83813 CF4BQ7 71562663 Ki > 300000 nM T83813 CRYO82 71562664 EC50 > 1000000 nM T83813 CQ0XA2 71562665 EC50 > 1000000 nM T83813 C5JX3D 71562666 EC50 > 1000000 nM T83813 CR9UC8 71562667 EC50 > 1000000 nM T83813 CJ8FA6 71652196 Ki = 12300 nM T83813 C5LY9W 71681897 EC50 = 16 nM T83813 CG34PR 71681898 EC50 = 193 nM T83813 CLA5P8 71681899 Ki = 1780 nM T83813 CG4V0A 71682216 EC50 = 70 nM T83813 CI46CW 71682217 EC50 = 77 nM T83813 CD87IN 71718791 Ki = 4786.3 nM T83813 C1ADL0 71720623 Ki = 309.03 nM T83813 C96DUR 71720624 Ki = 7200 nM T83813 C53MXL 71815503 IC50 = 1040 nM T83813 C9W2RC 72163104 Ki = 6.4 nM T83813 C3ATN5 72197484 IC50 = 1.98 nM T83813 C20HSN 72197485 IC50 = 13.3 nM T83813 CN8A5R 72197486 IC50 = 2.3 nM T83813 CL3BF7 72197668 EC50 = 9.2 nM T83813 C3TOA8 72205043 Ki = 8100 nM T83813 CO53SR 72205044 Ki = 2800 nM T83813 C5UN3D 72205045 Ki = 5100 nM T83813 CU4W5M 72205046 Ki = 5900 nM T83813 CZP67J 72205222 Ki = 7800 nM T83813 C8Z0NM 72550642 Ki = 26 nM T83813 CL6W2Q 72550645 Ki = 70 nM T83813 C78LYM 72698087 Ki > 10000 nM T83813 C63HPK 72698088 Ki = 980 nM T83813 C7W4RH 72734860 Ki = 200 nM T83813 CC6Q5R 72771081 Ki < 100 nM T83813 CC65OA 73213195 Ki > 10000 nM T83813 CW83DK 73213196 Ki > 10000 nM T83813 C0QCH3 73345916 IC50 = 8491 nM T83813 C2N9RL 73345917 IC50 = 242 nM T83813 CCNF45 73345918 IC50 > 10000 nM T83813 C6K8QF 73345919 IC50 = 5833 nM T83813 C9SN7B 73345920 IC50 = 5422 nM T83813 CXM8O2 73347306 IC50 = 700 nM T83813 C9X8GY 73347307 IC50 > 1000 nM T83813 C8LUG4 73347433 EC50 > 10000 nM T83813 C9GWD1 73347434 EC50 = 1200 nM T83813 CJ93GA 73347436 IC50 = 86.9 nM T83813 C3LO5H 73347437 IC50 = 29.4 nM T83813 C1FE6O 73347438 IC50 = 7787 nM T83813 CTG14R 73347439 IC50 > 10000 nM T83813 C8TCG6 73347440 IC50 = 148 nM T83813 CJP8E5 73347441 IC50 = 1179 nM T83813 CAZ9C2 73348087 IC50 = 156 nM T83813 C9RQM2 73348967 IC50 = 269 nM T83813 C5QDC1 73348968 IC50 = 5713 nM T83813 C4XAH0 73348969 IC50 = 3306 nM T83813 CJGF08 73348970 IC50 = 1300 nM T83813 CV31UL 73348972 IC50 = 7.8 nM T83813 C2CO5J 73350529 IC50 > 10000 nM T83813 C3B9NI 73350530 IC50 > 10000 nM T83813 C96DHM 73350531 IC50 > 10000 nM T83813 CZ7A4S 73350532 IC50 > 10000 nM T83813 C6LTU4 73350533 IC50 = 2588 nM T83813 CA20WC 73350534 IC50 = 3817 nM T83813 CKLH28 73350535 IC50 = 1500 nM T83813 CC8I7X 73351903 IC50 = 990 nM T83813 CG4M8P 73351905 IC50 > 1000 nM T83813 CZTE85 73352046 EC50 > 10000 nM T83813 CXZY13 73352047 IC50 = 1262 nM T83813 C6ZGY5 73352048 IC50 = 337 nM T83813 C0FWE9 73352049 IC50 = 416 nM T83813 CE09NW 73353508 EC50 = 9600 nM T83813 CRZ64E 73353509 IC50 = 779 nM T83813 CQOZ67 73353510 IC50 = 991 nM T83813 CZ5C3G 73353511 IC50 > 10000 nM T83813 CX4Q8N 73353512 IC50 = 4027 nM T83813 CBN58Q 73353513 IC50 = 1085 nM T83813 CAR7Z5 73354882 IC50 = 420 nM T83813 CY8S2M 73354999 IC50 > 10000 nM T83813 CN0P6A 73355000 IC50 > 10000 nM T83813 C23EYP 73355001 IC50 > 10000 nM T83813 CXM09L 73355002 EC50 = 2300 nM T83813 C61AQJ 73355003 IC50 = 333 nM T83813 CVFM82 73355005 IC50 > 10000 nM T83813 CNQ69I 73355006 IC50 > 10000 nM T83813 CQSJ15 73355007 IC50 = 494 nM T83813 CQZW41 73355008 IC50 = 836 nM T83813 CET52A 73356443 IC50 > 1000 nM T83813 CQAO31 73356563 EC50 = 2.6 nM T83813 CA6L7B 73356564 IC50 > 10000 nM T83813 CPG73S 73417116 EC50 = 2697 nM T83813 C8IDL3 75306277 Ki = 7.943 nM T83813 C1G6OH 76319284 EC50 = 76 nM T83813 C86INP 76322921 EC50 = 3 nM T83813 C4B1GO 76333762 EC50 = 0.4 nM T83813 C4RS7C 83753960 EC50 = 3.162 nM T83813 C70ZVB 86221574 Ki = 749 nM T83813 CJ9N5Q 86280005 Ki = 3.8 nM T83813 CCY5N2 86302554 Ki > 30000 nM T83813 CP76JG 88912137 Ki = 5000 nM T83813 CQ8I4E 90644510 EC50 > 10000 nM T83813 CWMU25 90644511 EC50 = 10 nM T83813 C1KX6L 90644512 EC50 > 10000 nM T83813 CYB8K4 90644513 Ki = 338.84 nM T83813 C2EZX4 90655112 Ki = 641 nM T83813 C6EZ3G 90655113 Ki = 503 nM T83813 CA08SW 90655114 Ki = 240 nM T83813 C42ELK 90655115 Ki = 89 nM T83813 C51ZIC 90655116 Ki > 1000 nM T83813 C4JOT3 90655117 Ki > 1000 nM T83813 CG2VY6 90655119 Ki = 3280 nM T83813 CV4H2G 90655120 Ki > 1000 nM T83813 CL3RP6 90655122 Ki > 1000 nM T83813 CVQC46 90655124 Ki > 1000 nM T83813 CB4Y0S 90655125 Ki > 1000 nM T83813 CH8YX5 90655126 Ki = 702 nM T83813 C8XT6K 90655127 Ki = 1280 nM T83813 C98YWT 90655128 Ki = 862 nM T83813 CBI6Y5 90664323 IC50 = 479 nM T83813 C2PV7O 90664324 IC50 = 88 nM T83813 CO4V5L 90664325 IC50 = 146 nM T83813 C2RW9Y 90664326 IC50 = 64 nM T83813 C6T1KX 90664327 IC50 = 50.8 nM T83813 C81IBN 90664328 IC50 = 189 nM T83813 C75ZUE 90664329 IC50 = 311 nM T83813 CM7HQ9 90664330 IC50 = 14.6 nM T83813 CA2BO3 90664449 IC50 = 64 nM T83813 C9ULV4 90664450 IC50 = 185 nM T83813 CH02GV 90664451 IC50 = 34.6 nM T83813 CIL2W9 90664452 IC50 = 1368 nM T83813 C7RT9G 90664453 IC50 = 76.6 nM T83813 C3AX1O 90664454 IC50 = 2221 nM T83813 CPGI68 90664459 IC50 = 233 nM T83813 CICD63 90664460 IC50 = 367 nM T83813 CBZT19 90664586 IC50 = 1509 nM T83813 C5HRY0 90664587 IC50 = 953 nM T83813 CG6V1D 90664589 IC50 = 459 nM T83813 C7W5SH 90664590 IC50 = 297 nM T83813 CNU6J8 90664598 IC50 = 39 nM T83813 CB95PE 90664599 IC50 = 551 nM T83813 CA68PB 90664600 IC50 = 62 nM T83813 C4MUI2 90664601 IC50 = 12.1 nM T83813 CA79EY 90664683 IC50 = 267 nM T83813 CHY82Q 90664697 IC50 = 535.2 nM T83813 CM0Y7P 90664699 IC50 = 383 nM T83813 CEF0R5 90664700 IC50 = 473 nM T83813 CR07QH 90664701 IC50 = 93.6 nM T83813 CZ69VH 90664702 IC50 = 774 nM T83813 CF4P3I 90664703 IC50 = 1454 nM T83813 CR7LX6 90664705 IC50 = 544 nM T83813 CNT10P 90664709 IC50 = 200 nM T83813 C35BTL 90664710 IC50 = 109 nM T83813 CDPV60 90664712 IC50 = 189 nM T83813 CG7D2H 90664713 IC50 = 139 nM T83813 CZJN57 90664814 IC50 = 855.9 nM T83813 CR87PO 90664815 IC50 = 229 nM T83813 CN7W8A 90664816 IC50 = 127 nM T83813 CI8B6Q 90664817 IC50 > 10000 nM T83813 CEN36Q 90664818 IC50 = 71 nM T83813 CJ73WT 90664819 IC50 = 284 nM T83813 C5AWS4 90664820 IC50 = 166.3 nM T83813 CL3AW1 90664821 IC50 = 526 nM T83813 C1C2HB 90664822 IC50 = 604 nM T83813 CQ4T3E 90664830 IC50 = 37.9 nM T83813 CTR58M 90664931 IC50 = 639 nM T83813 CP9SI1 90664949 IC50 = 155 nM T83813 CZ19LO 90664951 IC50 = 204 nM T83813 CLN9K2 90664952 IC50 = 113 nM T83813 CO5Y3C 90664958 IC50 = 235 nM T83813 C74XDT 90664959 IC50 = 106 nM T83813 CWQ18M 90664960 IC50 = 398 nM T83813 C07WIP 90664961 IC50 = 739 nM T83813 CHT7D5 90664962 IC50 = 66 nM T83813 C04UEP 90665072 IC50 = 661 nM T83813 CF90MU 90665073 IC50 = 663 nM T83813 C8YX4R 90665074 IC50 = 2239 nM T83813 CP5QO8 90665075 IC50 = 534 nM T83813 C3XIQ2 90665076 IC50 = 4375 nM T83813 CI8JU1 90665077 IC50 = 37.4 nM T83813 C67AXN 90665078 IC50 = 77 nM T83813 CQ95OT 90665079 IC50 = 323 nM T83813 C7JLM9 90665080 IC50 = 1365 nM T83813 CZHA09 90665086 IC50 = 110.6 nM T83813 C17EWV 90665087 IC50 = 61 nM T83813 CO46PW 90665091 IC50 = 198 nM T83813 CXJ62T 90665173 IC50 = 221 nM T83813 CYD25E 90665193 IC50 = 94.3 nM T83813 CG98QO 90665194 IC50 = 1506 nM T83813 C5PN4D 90665195 IC50 = 556.5 nM T83813 C7XIS2 90665197 IC50 = 476 nM T83813 CIJ5M0 90665200 IC50 = 140 nM T83813 C09JPN 90665201 IC50 = 109 nM T83813 C8BV5P 90665202 IC50 = 25.5 nM T83813 CACG19 90666899 Ki = 100 nM T83813 CODM50 90666903 Ki = 125.89 nM T83813 CRX16J 91884611 IC50 = 31.9 nM T83813 CUQ6V0 92042918 EC50 = 4.2 nM T83813 CGC29J 92042920 EC50 = 3.4 nM T83813 C02GRK 104697662 Ki = 3350 nM T83813 C5AFD3 112713234 EC50 = 1.995 nM T83813 C8V2SN 116887744 EC50 > 10000 nM T83813 CEMZ15 118464420 Ki = 156 nM T83813 CV2L6O 118464425 Ki = 1201 nM T83813 CFNG86 118464427 Ki = 1897 nM T83813 C5LFW4 118717221 Ki = 152 nM T83813 CES97Y 118722639 Ki = 79 nM T83813 CM3P7R 118722912 Ki > 1000 nM T83813 CP3QC2 118722913 Ki = 230 nM T83813 C1PG3C 118722914 Ki = 300 nM T83813 CR6E5D 118722915 Ki = 400 nM T83813 CDHS51 118727445 IC50 = 480 nM T83813 CZ1LD0 118727450 IC50 = 463 nM T83813 CU3X0M 118729231 Ki = 800 nM T83813 CNE49D 118729233 Ki = 7 nM T83813 CLD1Z7 118729234 Ki = 30 nM T83813 C4RDW3 118729235 Ki = 70 nM T83813 C47XHR 118729237 Ki = 78 nM T83813 C08FQG 118729239 Ki = 1000 nM T83813 CR0HA4 118729241 Ki = 520 nM T83813 CY36XK 118729243 Ki = 220 nM T83813 C1VK9B 118729245 Ki = 100 nM T83813 CVR67P 118729247 Ki = 70 nM T83813 CA2Y1F 118729249 Ki = 120 nM T83813 CE1IB3 118729250 Ki = 55 nM T83813 CI8WR2 118729251 Ki = 68 nM T83813 C4ML5K 118729252 Ki = 75 nM T83813 COCH98 118729253 Ki = 10 nM T83813 CQ7K5G 118729255 Ki = 120 nM T83813 C2LDI1 118729257 Ki = 10 nM T83813 COQ04B 118729259 Ki = 230 nM T83813 C9BG0R 118729261 Ki = 4 nM T83813 C63GWU 118729262 Ki = 200 nM T83813 CN24KA 118729263 Ki = 8 nM T83813 C7ZJ2F 118729265 Ki = 170 nM T83813 CL5W0J 118729267 Ki = 43 nM T83813 CN65HD 118729269 Ki = 200 nM T83813 C2B6YA 118729271 Ki = 30 nM T83813 CZ40RY 118729273 Ki = 1000 nM T83813 CE38GM 118729275 Ki = 5 nM T83813 CS9W7L 118729277 Ki = 50 nM T83813 C9LI7N 118729278 Ki = 290 nM T83813 C8TEX7 118729279 Ki = 2000 nM T83813 CW3R9X 118729280 Ki = 1600 nM T83813 C1D2KW 118733760 EC50 = 646 nM T83813 CJ1VX4 118733762 EC50 = 13 nM T83813 C2YQC3 118733764 EC50 = 1228 nM T83813 CSE5K7 118733766 EC50 = 103 nM T83813 C0QZ5N 118733767 EC50 = 683 nM T83813 C4JD7O 118733769 EC50 = 288 nM T83813 C8FZI7 118733776 EC50 = 1082 nM T83813 C4U6XR 118733778 EC50 = 251 nM T83813 C4V6FB 118733780 EC50 = 667 nM T83813 C1VB6N 118733781 EC50 = 183 nM T83813 CI9V0N 118733783 EC50 = 1762 nM T83813 C9HMQ0 118733785 EC50 = 244 nM T83813 CSZ6Q7 118733792 EC50 = 365 nM T83813 CQZ71R 118733794 EC50 = 63 nM T83813 C7MRW8 118733798 EC50 = 133 nM T83813 C7ZS0V 118733802 EC50 = 212 nM T83813 CWM78D 118733804 EC50 = 1127 nM T83813 C6VO5G 118733806 EC50 = 32 nM T83813 C7RUF2 118733808 EC50 = 914 nM T83813 CNH6K2 118733810 EC50 = 91 nM T83813 C0SH9U 118733812 EC50 = 1258 nM T83813 CXAZ36 118733814 EC50 = 206 nM T83813 C1CXD4 118733816 EC50 = 296 nM T83813 CSN70M 118733818 EC50 = 11 nM T83813 CD3E4N 118733819 EC50 = 157 nM T83813 CHFY98 118733821 EC50 = 985 nM T83813 CC4G2U 118733823 EC50 = 22 nM T83813 C98ZTE 118733825 EC50 = 514 nM T83813 C78OHM 118759078 EC50 > 10000 nM T83813 C2LW4N 122180957 EC50 = 218.78 nM T83813 CM1EW3 122180958 Ki = 2.512 nM T83813 C3LJ8I 122180959 Ki = 7.762 nM T83813 C4NA2C 122180960 Ki = 32.36 nM T83813 CP7DG4 122180961 Ki = 3.388 nM T83813 C6P9QO 122180962 Ki = 9.333 nM T83813 C8DSW3 122180963 Ki = 23.99 nM T83813 CS63HY 122180964 Ki = 66.07 nM T83813 CU4X9I 122180966 Ki = 70.79 nM T83813 CXQ4C1 122180967 Ki = 41.69 nM T83813 CX1N4V 122180968 Ki = 120.23 nM T83813 C90BHR 122180969 Ki = 154.88 nM T83813 CIL05K 122180970 Ki = 23.44 nM T83813 C0F9UN 122180971 Ki = 26.92 nM T83813 C2H8CK 122180972 Ki = 77.62 nM T83813 CKJ21N 122180973 Ki = 17.38 nM T83813 C6GI9R 122180974 Ki = 56.23 nM T83813 CBS6G1 122180975 Ki = 6.31 nM T83813 CDT10B 122180976 Ki = 4.677 nM T83813 C6A4CD 122180977 Ki = 20.89 nM T83813 CXL5V3 122183764 Ki = 44 nM T83813 CK3VT8 122183765 Ki = 14 nM T83813 C12TRH 122183771 Ki = 73 nM T83813 C06GQO 122183778 Ki = 1800 nM T83813 COP38R 122195446 IC50 = 51286.14 nM T83813 CJM64P 122195453 IC50 = 208929.61 nM T83813 CB91PC 122195454 IC50 = 269000 nM T83813 C7ODW3 122195524 Ki < 300 nM T83813 CV5L0S 122220128 Ki = 691.83 nM T83813 CLW53P 122483274 Ki = 1519 nM T83813 CO63ET 122483280 Ki = 1174 nM T83813 C4QM2E 124247485 Ki = 200 nM T83813 CCM0S8 126844990 EC50 = 4426 nM T83813 CWV9T8 127025170 Ki > 10000 nM T83813 CU67PG 127025781 Ki > 10000 nM T83813 C0SAG6 127025782 Ki > 10000 nM T83813 CG53JK 127025783 Ki > 10000 nM T83813 C7P8JY 127025784 Ki > 10000 nM T83813 CYG72J 127025785 Ki > 10000 nM T83813 CK92ZA 127025786 Ki > 1000 nM T83813 C3YG1L 127025787 Ki > 10000 nM T83813 C56JXR 127025788 Ki > 10000 nM T83813 CTBN56 127026052 Ki = 102.33 nM T83813 CL24NY 127026062 Ki > 10000 nM T83813 CC87HM 127026423 Ki = 140 nM T83813 C7Z0HG 127026424 Ki > 10000 nM T83813 CBHW31 127026425 Ki > 10000 nM T83813 C4CFA1 127026426 Ki > 1000 nM T83813 CQ85ZK 127026427 Ki > 10000 nM T83813 CBE56W 127026514 Ki = 588 nM T83813 C0SZI4 127026515 Ki = 1393 nM T83813 CAX87V 127026556 EC50 = 25 nM T83813 CH9JB5 127026860 EC50 = 223.87 nM T83813 C4PW9X 127026867 EC50 = 96 nM T83813 C3EA0C 127027022 Ki = 730 nM T83813 CU29SR 127027463 EC50 = 114.82 nM T83813 CW40RC 127028088 EC50 = 9.5 nM T83813 C7X4RJ 127028094 EC50 = 41.69 nM T83813 C7A8OC 127028095 EC50 = 3.8 nM T83813 CI1SF6 127028096 EC50 = 70.79 nM T83813 CGA51D 127028100 EC50 = 9.7 nM T83813 C90QPM 127028101 EC50 = 3.162 nM T83813 CALC05 127028403 EC50 = 107.15 nM T83813 C0SGM2 127028405 EC50 = 7.6 nM T83813 CE0T8G 127028406 EC50 = 3.162 nM T83813 C3H9NU 127028407 EC50 = 7.244 nM T83813 C8MC1I 127028408 EC50 = 8.7 nM T83813 CBU65F 127028421 EC50 = 18 nM T83813 C9YU1E 127028422 EC50 = 61 nM T83813 CPF1T5 127028423 EC50 = 0.95 nM T83813 CA9IP6 127028732 EC50 = 48.98 nM T83813 CG7OW2 127029036 EC50 = 36 nM T83813 CB8RL9 127029516 Ki > 10000 nM T83813 CC4U8R 127029581 EC50 = 23.99 nM T83813 C6O2SL 127034715 Ki = 194 nM T83813 CNO80F 127034729 Ki = 103 nM T83813 CZ61LK 127034966 EC50 > 5011.87 nM T83813 CA0SN5 127034967 EC50 > 5011.87 nM T83813 CQ0ZT9 127035062 Ki = 399 nM T83813 CW1KD7 127035063 Ki = 123 nM T83813 CO3W6A 127035064 Ki = 108 nM T83813 CTY04X 127035065 Ki = 206 nM T83813 CPM2B8 127035066 Ki = 273 nM T83813 CU49VE 127036186 Ki = 316.23 nM T83813 CP04WI 127036910 Ki = 1091 nM T83813 CG06BD 127036932 Ki = 204.17 nM T83813 CVW71O 127036953 Ki = 354.81 nM T83813 C0HLY8 127037059 Ki = 241 nM T83813 CZ6QR4 127037093 Ki = 690 nM T83813 CS9V0E 127048333 Ki = 79 nM T83813 CQM81O 127048334 Ki = 92 nM T83813 CJG5E2 127048335 Ki = 124 nM T83813 CUK40V 127048336 Ki = 68 nM T83813 CZS1L6 127049862 IC50 = 190 nM T83813 CZD91J 127049863 IC50 = 270 nM T83813 C6SP9O 127049979 Ki = 235 nM T83813 C1CB0Z 127049980 Ki = 219 nM T83813 C0JUA9 127049981 Ki = 224 nM T83813 C69RCG 127049982 Ki = 167 nM T83813 C0M9PE 127049983 Ki = 206 nM T83813 CI5XG2 127050282 Ki = 143 nM T83813 CX53AC 127050632 Ki = 614 nM T83813 CX5H1W 127051482 Ki = 126 nM T83813 C5ONG1 127051864 Ki = 4570.88 nM T83813 C6XR8U 127053028 Ki = 154 nM T83813 C6GC0F 129186534 IC50 = 90 nM T83813 C8KM6N 129186554 IC50 = 41.7 nM T83813 CEZT92 129186564 IC50 = 98.2 nM T83813 C10VDB 130431277 Ki = 5.4 nM T83813 CI1NF8 130431279 Ki = 22.4 nM T83813 CS8O4E 130431287 Ki = 55 nM T83813 C85MOW 130431289 Ki = 580 nM T83813 C2OH7B 130431291 Ki = 1780 nM T83813 CEQ43Y 130431295 Ki > 8900 nM T83813 CK64GU 130431296 Ki = 464 nM T83813 CYW0X2 130431314 Ki = 50 nM T83813 CDN26V 130431316 Ki = 113 nM T83813 CL64UW 130431317 Ki = 89 nM T83813 C8HE2O 130431318 Ki = 2190 nM T83813 CZ6S4T 130431319 Ki = 1110 nM T83813 C8ZHI7 130431325 Ki = 18.7 nM T83813 CF5SW8 130431328 Ki = 5670 nM T83813 CN9RZ3 130431329 Ki = 1260 nM T83813 CN70MW 130431337 Ki = 18.3 nM T83813 C4GF1U 130431342 Ki = 268 nM T83813 C2WI5R 130431351 Ki = 144 nM T83813 C1RI8Q 132060720 Ki = 2582 nM T83813 CY8B9L 132060743 Ki = 302 nM T83813 C7FM0U 132060763 Ki = 1338 nM T83813 CGHO19 132060770 Ki = 908 nM T83813 CT81OY 132060776 Ki = 1161 nM T83813 CFXL21 132060812 Ki = 1070 nM T83813 C7I5CQ 132118109 EC50 > 10000 nM T83813 CHB6K5 132118110 EC50 > 10000 nM T83813 CAVB41 132584404 Ki > 10000 nM T83813 CP26SI 132820207 EC50 = 25.12 nM T83813 CYBK37 132820208 EC50 = 1000 nM T83813 CEY94B 132820209 EC50 = 630.96 nM T83813 CC7PW1 132820210 EC50 = 79.43 nM T83813 CN08ZY 132820211 EC50 = 31.62 nM T83813 C78MPD 132820212 EC50 = 39.81 nM T83813 CYE4V1 134129923 Ki > 10000 nM T83813 C8O2EP 134130246 Ki = 1174.9 nM T83813 CM10CR 134132665 EC50 = 19.95 nM T83813 CQX4U3 134133064 Ki = 295.12 nM T83813 CGH25V 134133531 EC50 = 125.89 nM T83813 C0J2ML 134133604 Ki = 128 nM T83813 CP0E5M 134133632 Ki = 2028 nM T83813 CM0TS6 134133967 Ki = 675 nM T83813 CYRW09 134133994 EC50 > 10000 nM T83813 CP3J9C 134134314 Ki = 794.33 nM T83813 CZ8HL0 134134668 Ki = 703 nM T83813 C6G4CW 134135745 Ki = 190 nM T83813 CZ0RN8 134136722 EC50 = 125.89 nM T83813 CBOH57 134136932 EC50 = 125.89 nM T83813 CS1HT4 134137343 EC50 = 3.981 nM T83813 CE93ZP 134137441 EC50 = 63.1 nM T83813 CEU49D 134137640 EC50 > 1000 nM T83813 C9A6KG 134138183 Ki = 371 nM T83813 C5JP1R 134138627 EC50 = 158.49 nM T83813 CH0FX4 134138769 Ki = 270 nM T83813 C0XHJ2 134139670 EC50 = 63.1 nM T83813 CR7C9U 134139964 Ki = 0.631 nM T83813 CNSB82 134141050 Ki = 2580 nM T83813 C86RBW 134141127 EC50 = 6.31 nM T83813 CLW86T 134141354 Ki = 346.74 nM T83813 C4ECW0 134141640 EC50 = 199.53 nM T83813 C68AXD 134141831 Ki = 84 nM T83813 CCS9A1 134142903 Ki = 0.631 nM T83813 CJFV62 134143302 Ki = 1700 nM T83813 C08RJA 134143536 Ki = 298 nM T83813 C5L9BD 134143752 Ki = 3.9 nM T83813 CV8IR0 134143977 Ki = 0.3981 nM T83813 C1NDF5 134144277 EC50 = 100 nM T83813 CR5L4K 134144303 Ki = 611 nM T83813 C71PIY 134144970 Ki = 205 nM T83813 CC9P2T 134146194 Ki = 501 nM T83813 C8C3GJ 134146228 EC50 = 10 nM T83813 C19LRO 134146585 Ki = 4300 nM T83813 CUQ0F6 134147456 EC50 = 0.1995 nM T83813 CZPS45 134148291 EC50 = 19.95 nM T83813 C7S5RQ 134149008 Ki = 8000 nM T83813 CBU81N 134149168 Ki = 1679 nM T83813 COUJ52 134149355 Ki = 0.7943 nM T83813 CAO9T6 134150123 Ki = 1350 nM T83813 CM31CH 134150311 EC50 > 1000 nM T83813 CLU34D 134151427 Ki = 1174.9 nM T83813 CFV6S8 134151626 EC50 = 19.95 nM T83813 C8PT9W 134152052 Ki = 269 nM T83813 C73ISY 134152157 Ki = 251 nM T83813 CL0G3W 134152924 EC50 = 0.3162 nM T83813 CT16QG 134153263 EC50 = 1258.93 nM T83813 CB6M5Y 134153538 Ki = 812.83 nM T83813 CP41RT 134154065 Ki = 4.1 nM T83813 C79TEI 134154068 Ki = 758.58 nM T83813 CMJ1U3 134154387 Ki = 2884.03 nM T83813 C4VGJ5 134154679 Ki = 329 nM T83813 C79QLN 134155460 Ki > 10000 nM T83813 CZFB29 134155462 Ki = 8100 nM T83813 CE64VO 134155579 EC50 = 25.12 nM T83813 CZJ15H 134155852 Ki = 0.3162 nM T83813 C87HWQ 134155992 EC50 = 19.95 nM T83813 CVR87Q 134156222 Ki = 4234 nM T83813 C7UOJ8 134156506 Ki = 672 nM T83813 C1IF0S 134156657 EC50 = 3.162 nM T83813 C5UQW2 134157367 Ki = 2310 nM T83813 C3BDA6 134157788 Ki = 8500 nM T83813 CF7EV5 134265590 EC50 = 329 nM T83813 CL5FW8 134265616 EC50 = 0.108 nM T83813 CR06XB 134265618 EC50 = 12.3 nM T83813 CNA08H 134265620 EC50 = 0.116 nM T83813 C46YNU 134265622 EC50 = 5.84 nM T83813 CA5PX2 134265627 EC50 = 0.19 nM T83813 CAS9Z4 134265663 EC50 = 1.14 nM T83813 CW3I6K 134265665 EC50 = 1.17 nM T83813 CVY5G8 134265675 EC50 = 7.5 nM T83813 C6SLE4 134265705 EC50 = 93.4 nM T83813 C8WAR6 134265732 EC50 = 1.33 nM T83813 C6N8GM 135367405 Ki = 296 nM T83813 C6LU0C 135367816 Ki = 1099 nM T83813 CD2TH9 135367820 Ki = 785 nM T83813 C5AMD9 135367857 Ki = 20 nM T83813 CGBW93 135410312 Ki = 11.22 nM T83813 C8WL0I 135449090 Ki = 10000 nM T83813 CVE08Y 135458392 Ki = 235 nM T83813 CP7HN4 135458393 Ki = 401 nM T83813 CS8XJ6 135458394 Ki = 94 nM T83813 C9B7XA 135458410 Ki = 162 nM T83813 CFV9A3 135458427 Ki = 2145 nM T83813 CKX4N8 135458428 Ki = 1658 nM T83813 CTE23K 135464118 Ki = 35 nM T83813 C7DF4S 135464159 Ki = 67.61 nM T83813 CB53EI 135465870 Ki = 2354 nM T83813 C7AGR0 135474338 Ki = 1916 nM T83813 CP9XN7 135500023 Ki = 181.97 nM T83813 C34FXW 135501716 Ki = 4348 nM T83813 C0H9YX 135507495 Ki = 50.12 nM T83813 C1CZ9M 135514796 Ki = 349 nM T83813 C6I9RK 135516645 Ki = 112.2 nM T83813 CQI23C 135516796 Ki = 151.36 nM T83813 C3FV9I 135527031 Ki = 346.74 nM T83813 CNI90F 135797785 Ki = 580 nM T83813 C03HVY 135846955 Ki = 10000 nM T83813 CQCT18 135846958 Ki = 3883 nM T83813 CE4QG5 135846981 Ki = 10000 nM T83813 C3UB7L 135846982 Ki = 10000 nM T83813 CA1M8B 135966709 Ki = 970 nM T83813 CUKO20 136020617 Ki > 10000 nM T83813 COF0U5 136020618 Ki = 1600 nM T83813 CF89JI 136030596 Ki > 10000 nM T83813 CE8GB9 136030693 Ki > 10000 nM T83813 C65VFI 136030744 Ki > 10000 nM T83813 CJ45EW 136044083 EC50 = 1460 nM T83813 COIX80 136054961 Ki > 10000 nM T83813 C19GLK 136116062 Ki = 675 nM T83813 CUG28I 136117980 Ki = 810 nM T83813 CA3JC8 136118613 Ki = 1698 nM T83813 CQ2GP6 136118614 Ki = 1271 nM T83813 C6R4IC 136118615 Ki = 10000 nM T83813 CS0JL5 136118616 Ki = 320 nM T83813 C8RH6M 136118617 Ki = 1078 nM T83813 CN4U6K 136118618 Ki = 2275 nM T83813 CHWC38 136118619 Ki = 2208 nM T83813 C5UDW3 136118620 Ki = 2762 nM T83813 C8I6UN 136118621 Ki = 3013 nM T83813 CV4E6W 136118635 Ki = 1870 nM T83813 C0UH1B 136118638 Ki = 885 nM T83813 C6G4AY 136118639 Ki = 2094 nM T83813 C40VES 136118640 Ki = 4367 nM T83813 C43JTG 136118647 Ki = 970 nM T83813 CLH0V9 136118648 Ki = 80 nM T83813 C76XEJ 136118649 Ki = 426 nM T83813 CN0V5C 136118650 Ki = 980 nM T83813 CR72MQ 136118651 Ki = 678 nM T83813 CD7OE2 136118652 Ki = 2339 nM T83813 CG5TX8 136118653 Ki = 1343 nM T83813 CCHM67 136118657 Ki = 10000 nM T83813 C0W1TM 136118658 Ki = 1856 nM T83813 C40LYH 136118659 Ki = 2430 nM T83813 CZ7C3Y 136118660 Ki = 1239 nM T83813 C42FCS 136118661 Ki = 6470 nM T83813 CR3DK1 136118716 Ki = 604 nM T83813 CON04G 136118728 Ki = 201 nM T83813 COX1F8 136118729 Ki = 841 nM T83813 CY5GU4 136118730 Ki = 2013 nM T83813 C0R5PV 136118732 Ki = 4129 nM T83813 C08PTG 136123530 IC50 = 589 nM T83813 CB12QP 136152964 Ki = 351.7 nM T83813 CFX06E 136152966 Ki = 233 nM T83813 C37YXA 136152971 Ki = 121 nM T83813 CY0C1X 136152972 Ki = 238 nM T83813 CSNE17 136179514 Ki = 144.54 nM T83813 CT0ZC8 136179515 Ki = 43.65 nM T83813 CAE39V 136188797 Ki > 10000 nM T83813 CLAP52 136259032 Ki > 10000 nM T83813 CGS61F 137553161 Ki = 238 nM T83813 CBX2V5 137631812 EC50 = 17 nM T83813 CQO58W 137632042 EC50 = 381 nM T83813 CDQ6X3 137632069 EC50 = 58 nM T83813 CS5K0I 137632108 EC50 = 229.09 nM T83813 C64KPN 137632218 EC50 = 119 nM T83813 C96DFN 137632449 EC50 = 2550 nM T83813 CMO30D 137633009 EC50 = 1804 nM T83813 C5ZL0C 137633983 EC50 = 18 nM T83813 CATU84 137634233 EC50 >= 4100 nM T83813 CXCJ60 137634432 EC50 > 10000 nM T83813 C9M3RV 137635151 EC50 = 524.81 nM T83813 C94MFJ 137635172 EC50 = 1040 nM T83813 C5N4PR 137635711 EC50 = 38 nM T83813 CJT0A2 137635932 EC50 = 4600 nM T83813 CPQ34V 137636430 EC50 = 2780 nM T83813 CQ71WO 137636435 EC50 = 1272 nM T83813 C8Z1XW 137636480 EC50 = 8.913 nM T83813 C4OT7C 137637069 EC50 = 1600 nM T83813 CTD64R 137637165 EC50 = 43 nM T83813 CK29VL 137637650 EC50 = 530 nM T83813 C71BUE 137637880 EC50 = 245 nM T83813 C56GTL 137638508 EC50 = 13 nM T83813 CM0DJ5 137638903 EC50 = 766 nM T83813 CBK0I8 137639266 Ki = 258 nM T83813 CK8UC2 137639485 EC50 = 24 nM T83813 CI5Q2P 137639497 Ki = 430 nM T83813 CEQ68W 137639630 EC50 = 41 nM T83813 CPQ83I 137639705 EC50 = 3850 nM T83813 C5KX6V 137640062 EC50 = 23.5 nM T83813 CKJD12 137640272 EC50 = 228 nM T83813 CPK8A0 137640608 EC50 = 1621.81 nM T83813 C62QAM 137640945 EC50 = 776.25 nM T83813 C90GKM 137641125 EC50 = 7 nM T83813 CUQ8F5 137641376 EC50 = 1520 nM T83813 C6P9FW 137642149 EC50 = 501 nM T83813 C4HJ1N 137642593 EC50 = 549.54 nM T83813 CO6J9Q 137642857 EC50 = 12 nM T83813 CX65BH 137643424 EC50 = 870.96 nM T83813 CPL0K5 137643658 EC50 = 1870 nM T83813 C1ZP9R 137643846 EC50 = 28 nM T83813 CIKD85 137644487 EC50 > 10000 nM T83813 CRGN16 137644935 EC50 = 399 nM T83813 CSO38A 137645024 EC50 = 1697 nM T83813 CRU20V 137645667 EC50 = 315 nM T83813 CA7P4F 137645674 EC50 = 12 nM T83813 CUR7T5 137645858 EC50 = 1522 nM T83813 C5Q6DL 137646111 EC50 = 679 nM T83813 CPI68E 137646281 Ki = 159 nM T83813 C4YE8H 137646603 EC50 = 120 nM T83813 C9EYB1 137646716 EC50 = 47 nM T83813 C2O1XW 137646874 EC50 > 10000 nM T83813 C6C3IK 137646921 EC50 = 6 nM T83813 CN5R7Q 137647004 EC50 = 30 nM T83813 CD2TE0 137647007 EC50 = 13 nM T83813 C5Y0FG 137647246 EC50 = 129 nM T83813 CU6V5W 137647439 EC50 = 22.91 nM T83813 CRC30Z 137647475 EC50 = 95 nM T83813 CA48GB 137647635 EC50 = 5 nM T83813 CQA0B2 137647926 EC50 = 15 nM T83813 CR64OK 137648428 EC50 = 1860 nM T83813 C4HX6J 137648810 EC50 >= 3460 nM T83813 C2VBA0 137649655 EC50 = 670 nM T83813 C1GZV3 137650863 EC50 = 615 nM T83813 CXV3D7 137651249 EC50 = 729 nM T83813 C71DPJ 137651253 EC50 = 1200 nM T83813 CWG87E 137651507 Ki = 395 nM T83813 C1SY4J 137651715 EC50 = 450 nM T83813 CTE69H 137652480 EC50 = 6 nM T83813 CY59NZ 137652713 EC50 = 14 nM T83813 CPFG35 137653140 EC50 = 308 nM T83813 CR9F3Q 137653203 Ki = 3240 nM T83813 C04XYN 137653567 IC50 = 2.69 nM T83813 CC12VB 137653689 EC50 = 3100 nM T83813 CKT1F5 137654351 EC50 = 334 nM T83813 CS1Y8F 137654798 EC50 = 16 nM T83813 CZ50SL 137654926 EC50 = 63 nM T83813 CJMR75 137655187 EC50 = 407.38 nM T83813 C53QIZ 137655324 EC50 = 2.399 nM T83813 CHI8M2 137655535 EC50 = 190 nM T83813 CB20MW 137655657 EC50 = 433 nM T83813 C91UBP 137655705 EC50 = 47 nM T83813 C1PKE6 137655741 EC50 = 95 nM T83813 CKW87Y 137655846 EC50 = 1032 nM T83813 CZ82HF 137655858 EC50 = 2600 nM T83813 C60XIF 137655882 EC50 = 27 nM T83813 C17NVY 137656030 EC50 = 291 nM T83813 CL8RT7 137656524 EC50 > 10000 nM T83813 C1SX4C 137656726 EC50 = 302 nM T83813 CCKP95 137657310 EC50 = 120.23 nM T83813 CKQ7Y9 137658074 EC50 = 4528 nM T83813 C0OI2B 137658246 EC50 = 369 nM T83813 CH9R5V 137658409 EC50 = 576 nM T83813 CBK37P 137658537 EC50 = 524.81 nM T83813 C3JG5Z 137659281 EC50 = 59 nM T83813 CAM68B 137660072 EC50 = 20 nM T83813 C5Q9CM 137660307 EC50 = 102.33 nM T83813 C3UHP5 137660422 EC50 = 68 nM T83813 C6SHF4 137661018 EC50 > 10000 nM T83813 CO2TV7 137661051 EC50 = 501.19 nM T83813 C0YZF2 137661221 EC50 = 25 nM T83813 CEJ38Q 137661378 EC50 = 12.88 nM T83813 C8JH6R 137661673 EC50 = 2 nM T83813 CN52AG 137662193 EC50 = 320 nM T83813 C7KC3T 145963830 Ki = 770 nM T83813 CEN94V 145963961 IC50 = 70 nM T83813 CHDN35 145964150 Ki = 3200 nM T83813 C1KH2E 145964159 Ki = 140 nM T83813 C1B8QW 145964299 IC50 = 63 nM T83813 C12OVL 145965034 Ki > 10000 nM T83813 CKO51D 145965628 Ki = 1400 nM T83813 C5W4LM 145965940 Ki = 2400 nM T83813 C4EQ9C 145966293 EC50 = 33.6 nM T83813 CLM10C 145966333 IC50 = 346 nM T83813 C81VUO 145967771 Ki = 2200 nM T83813 CJS56K 145967795 Ki > 10000 nM T83813 CQJ5O8 145971635 Ki = 3600 nM T83813 C7BVC1 145972374 Ki = 820 nM T83813 C79TNE 145972796 Ki = 1900 nM T83813 C6XIN0 145974114 Ki > 10000 nM T83813 CD8ZL6 145974750 Ki > 10 nM T83813 C6PH4F 145975226 Ki = 880 nM T83813 C71CYU 145975946 Ki = 1700 nM T83813 C2TN8W 145976085 Ki = 1200 nM T83813 C7L9DG 145976983 Ki = 2300 nM T83813 C6BFY7 145977338 Ki > 10000 nM T83813 C0Y6QO 145977799 Ki = 750 nM T83813 C3BI1R 145978113 Ki = 35000 nM T83813 CQU8R0 145978665 Ki = 5400 nM T83813 C6AV9G 145978819 Ki = 2200 nM T83813 C6RV3M 145979282 Ki = 9 nM T83813 CUM97N 145979585 Ki = 285 nM T83813 CV8K7E 145979689 Ki > 10000 nM T83813 C87MSW 145980271 Ki = 1126 nM T83813 C8I7QL 145980875 Ki = 2548 nM T83813 CM7D2G 145981162 Ki = 145 nM T83813 C1YJ0P 145981769 Ki = 160 nM T83813 CH5A3J 145982070 Ki > 10000 nM T83813 C9R8FK 145982167 Ki = 580 nM T83813 C6I5AL 145982333 Ki = 15 nM T83813 CO7R2A 145983175 Ki = 8 nM T83813 C1DW4U 145983928 IC50 = 341 nM T83813 CF8T9A 145983929 Ki = 1600 nM T83813 CM2C9Z 145986330 Ki = 72 nM T83813 C7VJ9I 145986532 Ki = 61 nM T83813 C3D6RX 145986700 Ki > 10000 nM T83813 CNJH37 145986752 Ki = 740 nM T83813 C7U2SG 145987794 Ki = 60 nM T83813 C7C6XZ 145988269 Ki > 10000 nM T83813 C86XQR 145988313 Ki = 473 nM T83813 CUGO10 145988693 Ki = 402 nM T83813 CC83DQ 145988741 Ki = 200 nM T83813 C5Q8HG 145988801 Ki = 180 nM T83813 CH04CY 145990308 Ki = 42 nM T83813 CRH4A6 145990662 Ki > 10000 nM T83813 CMJ46R 145990794 IC50 = 188 nM T83813 C2NF4G 145991111 Ki = 400 nM T83813 C73PGR 145991966 Ki = 100 nM T83813 CCP2U1 145992489 Ki = 1603 nM T83813 CU94SI 145992795 Ki > 10000 nM T83813 C9PS8N 145993117 IC50 = 606 nM T83813 CX8HD4 145993188 Ki > 10000 nM T83813 CZLY96 145993214 Ki = 340 nM T83813 C0Z6YX 145993493 IC50 = 400 nM T83813 C43VNT 145993566 Ki = 190 nM T83813 C6P3SR 153287553 Ki > 10000 nM T83813 CV9G7Z 153287572 Ki = 2511.89 nM T83813 CO85KL 153287574 Ki = 3981.07 nM T83813 CZ53NG 153605599 Ki = 1450 nM T83813 CU4H6L 155512064 Ki > 10000 nM T83813 CCD9N1 155512086 Ki = 1320 nM T83813 C7Q1RY 155512645 EC50 = 110 nM T83813 C2J0BS 155513179 Ki = 450 nM T83813 CHXY56 155513802 Ki = 165 nM T83813 CL5G9Q 155513837 Ki = 513 nM T83813 CK9YN0 155514430 Ki = 1000 nM T83813 CH34RK 155514798 Ki = 125.9 nM T83813 CUE5J3 155515907 Ki = 53 nM T83813 CV12SD 155516041 Ki = 417 nM T83813 CJ98ZK 155516236 Ki = 412.1 nM T83813 C7GK1V 155516859 EC50 = 5245 nM T83813 C9ZAW0 155517266 Ki = 1259 nM T83813 CUSA24 155519891 Ki = 1584.89 nM T83813 C0F8YT 155521278 Ki = 550 nM T83813 CV7IG5 155522663 Ki = 495.4 nM T83813 C2H3JL 155523073 Ki = 57.5 nM T83813 CQA76T 155523112 Ki = 132 nM T83813 C3E9DJ 155523127 Ki = 1339 nM T83813 CVQ68Y 155523770 Ki = 63.1 nM T83813 COH1Q5 155524191 Ki = 427 nM T83813 CW7NT8 155524423 Ki = 105 nM T83813 CQX27T 155525357 Ki = 136 nM T83813 CGS21U 155525549 Ki > 10000 nM T83813 CW65KS 155525705 Ki = 85 nM T83813 C65WSA 155527636 Ki = 80 nM T83813 CRF1A0 155527638 EC50 = 4.169 nM T83813 C8QF4Y 155529999 Ki = 200 nM T83813 CV6ST2 155531084 Ki = 338 nM T83813 CX43DV 155532107 EC50 = 2.754 nM T83813 CKZ35G 155532475 Ki = 2171 nM T83813 CZA89B 155533824 Ki = 4 nM T83813 CQ12KS 155533996 Ki = 179 nM T83813 C8AX5N 155534186 Ki = 2362 nM T83813 C3JPS4 155534559 EC50 = 309.03 nM T83813 COT9U8 155535203 Ki = 8320 nM T83813 CGZ5T8 155535272 Ki = 222 nM T83813 CHP2Z9 155535866 Ki = 137 nM T83813 C7OIP3 155535969 EC50 = 4073.8 nM T83813 CB79ZW 155536080 Ki = 2511.89 nM T83813 CIUS98 155536619 Ki = 2350 nM T83813 CVFD68 155537516 Ki = 1122 nM T83813 C13CSU 155537907 Ki = 274 nM T83813 C0A9WG 155539425 EC50 = 220 nM T83813 C4FJL0 155539960 EC50 = 598 nM T83813 C72KHI 155540514 EC50 = 12 nM T83813 C1JM5R 155540523 Ki = 343 nM T83813 CVK2M9 155543189 Ki = 136 nM T83813 C4ANI0 155543691 Ki = 44.7 nM T83813 CMT60C 155543832 Ki = 1750 nM T83813 C08FTE 155544239 Ki = 97.7 nM T83813 CGU5M0 155544723 Ki > 10000 nM T83813 C7MCZ0 155546478 Ki = 68 nM T83813 CSX3M0 155548666 EC50 = 288.4 nM T83813 C9BAV3 155549312 Ki = 250 nM T83813 C7KWB9 155550387 Ki = 32 nM T83813 CN6I4P 155550431 Ki = 219 nM T83813 C6N9PG 155550640 Ki = 238 nM T83813 CG7NR9 155550756 Ki = 898 nM T83813 CN39VC 155551164 EC50 = 229 nM T83813 C82QWR 155551173 Ki = 49 nM T83813 CG70XQ 155552591 Ki = 284 nM T83813 CF0W4K 155552683 Ki = 1190 nM T83813 C0DQ3Z 155552695 Ki = 17.2 nM T83813 CQ25NV 155553234 EC50 = 1064 nM T83813 CD5LC6 155554006 Ki = 85.1 nM T83813 C0PBT3 155555147 Ki > 10000 nM T83813 C36SYJ 155558844 Ki = 49 nM T83813 C5L8HB 155560629 EC50 = 5.012 nM T83813 C9LV7U 155561048 EC50 = 789 nM T83813 C7OZM6 155561446 Ki = 138 nM T83813 CSK27Q 155561712 Ki = 24 nM T83813 CLS45N 155562708 EC50 = 70 nM T83813 C9P7AU 155562772 Ki = 120 nM T83813 C4N9GU 155563428 Ki = 89 nM T83813 C8YPA7 155564299 EC50 = 7.943 nM T83813 C0UN4V 155564747 Ki = 203 nM T83813 CR12DI 155565189 IC50 > 100000 nM T83813 CMH8I1 155565768 Ki = 1308 nM T83813 CBI7N3 155566272 Ki = 1460 nM T83813 CK20WA 155566662 Ki = 535 nM T83813 C6DPR8 155566974 Ki = 61.7 nM T83813 CPW8M5 155567457 Ki = 1100 nM T83813 C5A6YM 155567869 Ki = 123 nM T83813 CV24CW 155568676 Ki = 106 nM T83813 C42JKO 155569198 Ki = 50.1 nM T83813 C3N9VU 10251906 Ki = 2 nM T83813 CP9TR0 10324985 Ki = 99.6 nM T83813 CQ1LV7 135508617 Ki = 1265 nM T83813 CGK7B1 135511529 Ki = 4778 nM T83813 C96JQU 135860585 Ki = 46 nM T83813 C6ZSL7 136016497 Ki = 5230 nM T83813 CE2J8F 136016507 Ki = 2114 nM T83813 CRKP76 136016509 Ki = 2454 nM T83813 CWKJ21 136016511 Ki = 166 nM T83813 CKM28Y 136016513 Ki = 8323 nM T83813 CB2VD8 44241743 Ki = 173 nM T83813 D00APD 15124 Ki = 6800 nM T83813 D00AVR 135476741 Ki = 10000 nM T83813 D00BWZ 10823903 Ki = 1258.93 nM T83813 D00DHV 2760428 Ki = 113 nM T83813 D00EMF 3644637 Ki = 1 nM T83813 D00FHZ 124007 IC50 = 6400 nM T83813 D00GOY 6604042 Ki = 24 nM T83813 D00LXH 10753358 Ki = 3.981 nM T83813 D00NST 44452811 Ki = 0.2 nM T83813 D00OBS 44559159 Ki = 4630 nM T83813 D00OCV 44404892 Ki = 539 nM T83813 D00PEU 4847 Ki = 60 nM T83813 D00YVE 10219723 EC50 = 2.3 nM T83813 D01BGW 11708275 Ki = 1.5 nM T83813 D01CGM 3033677 Ki = 40 nM T83813 D01CXD 10398175 Ki = 43 nM T83813 D01FOM 16768198 Ki = 127 nM T83813 D01KAX 135453290 Ki = 3 nM T83813 D01NTM 11264955 Ki = 3.2 nM T83813 D01PYU 9821248 Ki = 2400 nM T83813 D01SJL 135509961 Ki = 1.2 nM T83813 D01TSX 9840090 Ki = 4 nM T83813 D01WNO 21868720 Ki = 560 nM T83813 D01WWC 16573 Ki > 950 nM T83813 D01XZI 10015055 Ki = 430 nM T83813 D02ESW 107992 EC50 = 28 nM T83813 D02UWB 1809 IC50 = 588.84 nM T83813 D02YNH 9901086 EC50 = 0.11 nM T83813 D02YSX 197033 Ki = 75.86 nM T83813 D03DET 10287730 Ki = 3162.28 nM T83813 D03DLZ 6089 Ki = 33 nM T83813 D03JOX 11311147 IC50 > 10000 nM T83813 D03ZHB 44455973 Ki = 380 nM T83813 D04AQE 1833 Ki = 45 nM T83813 D04AZE 3277600 Ki = 1513.56 nM T83813 D04QRS 27559 EC50 = 7.7 nM T83813 D04TPO 16006492 Ki = 152 nM T83813 D04UCV 14595512 Ki = 1460 nM T83813 D04VXP 2794808 Ki = 22 nM T83813 D04YCJ 135399866 Ki = 1 nM T83813 D05EQG 5265 Ki = 630.96 nM T83813 D05FKE 46228441 Ki = 378 nM T83813 D05GDP 599482 Ki > 10000 nM T83813 D05JIO 9859429 Ki = 32 nM T83813 D05NWH 443390 Ki = 1 nM T83813 D05RKH 46228435 Ki = 156 nM T83813 D05SWY 44404899 Ki = 12.6 nM T83813 D05XGR 6918647 Ki = 1000 nM T83813 D05ZUX 44207909 Ki >= 1000 nM T83813 D06ABJ 11492162 Ki = 82 nM T83813 D06QGD 11357862 IC50 > 10000 nM T83813 D06VDN 443391 IC50 = 0.7 nM T83813 D07DQO 44250365 IC50 = 542 nM T83813 D07ETF 9838960 Ki = 150 nM T83813 D07GBV 10091189 Ki = 79 nM T83813 D07GQP 11477180 Ki = 47 nM T83813 D07LHD 44404907 Ki = 2182 nM T83813 D07LRJ 5312149 Ki = 530 nM T83813 D07LVT 16726095 Ki = 4357 nM T83813 D07XTU 1229 Ki = 1.82 nM T83813 D07ZOP 11470616 IC50 > 10000 nM T83813 D08BCF 5011 IC50 = 61.66 nM T83813 D08CKM 9863250 Ki < 5011.87 nM T83813 D08CZT 9882067 Ki = 400 nM T83813 D08DOG 25130235 Ki = 3000 nM T83813 D08EFH 36906 Ki = 8.3 nM T83813 D08FUK 10845306 Ki = 63 nM T83813 D08GJS 44404906 Ki = 126 nM T83813 D08JCU 44439386 Ki = 200 nM T83813 D08OFG 11177588 Ki = 340 nM T83813 D08VGJ 9904281 Ki = 208 nM T83813 D08YZM 18008465 EC50 = 755 nM T83813 D08ZWM 4980 EC50 = 30 nM T83813 D09BNS 439280 EC50 = 0.18 nM T83813 D09HFT 44439376 Ki > 4000 nM T83813 D09HJL 10331436 Ki = 3.4 nM T83813 D09OYA 2107 Ki = 6.6 nM T83813 D09PIN 3378093 Ki = 630.96 nM T83813 D09RPR 16737207 Ki > 10000 nM T83813 D09WIL 10028436 Ki = 269.15 nM T83813 D0A6LB 46228433 EC50 = 25 nM T83813 D0AP6N 44404886 Ki = 4.4 nM T83813 D0B3WX 5475158 Ki = 200 nM T83813 D0C1SE 14595509 Ki = 4780 nM T83813 D0C5XQ 1832 Ki = 42 nM T83813 D0CK9K 6918513 IC50 = 5500 nM T83813 D0D3YN 1238 Ki = 0.57 nM T83813 D0DY5G 443389 Ki = 2.512 nM T83813 D0E3AL 56597938 Ki = 0.6 nM T83813 D0E6NW 9859257 EC50 = 4.5 nM T83813 D0F0IA 11301655 Ki > 2000 nM T83813 D0F1FN 15893127 Ki = 720 nM T83813 D0F5WP 135520431 Ki = 9.6 nM T83813 D0F6CD 5202 EC50 = 0.09 nM T83813 D0FF6S 16038374 IC50 > 10000 nM T83813 D0FL1D 9842124 Ki = 2000 nM T83813 D0FU5E 10220053 Ki > 1000 nM T83813 D0G7LE 10991121 Ki = 46 nM T83813 D0G7QT 10131112 IC50 = 450 nM T83813 D0G8CV 9954003 Ki = 199.53 nM T83813 D0H3WJ 44435193 Ki = 390 nM T83813 D0H5XR 3045225 Ki = 0.89 nM T83813 D0H7PC 6918553 Ki > 5011.87 nM T83813 D0H9QG 5312148 Ki < 15848.93 nM T83813 D0I9KV 11220599 IC50 > 10000 nM T83813 D0I9RW 135427931 Ki = 4.8 nM T83813 D0J1VB 10966027 Ki = 14 nM T83813 D0J2ID 10730997 Ki = 50 nM T83813 D0J2UA 135433933 Ki = 330 nM T83813 D0J2YB 23631116 Ki > 1000 nM T83813 D0J6JT 1355 EC50 = 7.943 nM T83813 D0J8RI 9964324 Ki = 6.3 nM T83813 D0K5NZ 68848 Ki = 0.92 nM T83813 D0K6VR 44287208 Ki = 520 nM T83813 D0KU6D 10679289 Ki = 3.981 nM T83813 D0KV4G 15887436 IC50 = 24 nM T83813 D0L5MW 181743 Ki = 1069 nM T83813 D0L8MR 4076 Ki = 302.8 nM T83813 D0M1YU 10198431 Ki = 1.6 nM T83813 D0M3PV 133633 Ki = 6570 nM T83813 D0M5ZE 5311416 Ki = 1584.89 nM T83813 D0N8YG 135414348 Ki = 3.6 nM T83813 D0ND5D 10493741 Ki = 2000 nM T83813 D0NM6R 135412764 Ki = 3500 nM T83813 D0O3GF 1220 Ki = 7250 nM T83813 D0O3GQ 11849796 Ki = 150 nM T83813 D0O5KK 44451373 Ki = 23 nM T83813 D0OG0R 10337743 IC50 = 644 nM T83813 D0PC7A 10106214 Ki = 30 nM T83813 D0Q3OK 9855823 Ki = 7.9 nM T83813 D0Q4AQ 46228424 Ki = 207 nM T83813 D0Q9FU 10330734 Ki = 1 nM T83813 D0Q9KP 44452853 Ki = 43 nM T83813 D0R3GW 10296414 Ki < 7943.28 nM T83813 D0R5WB 9817960 Ki = 268 nM T83813 D0R8VT 44404883 Ki = 7 nM T83813 D0RC9T 9795587 Ki = 89 nM T83813 D0S0XK 9863146 IC50 = 1862.09 nM T83813 D0SP2J 10257 Ki = 70 nM T83813 D0T2RY 9948320 Ki >= 1000 nM T83813 D0T7RY 9813197 Ki = 8.8 nM T83813 D0T8UR 44404904 Ki = 87 nM T83813 D0U5HQ 44287445 Ki = 490 nM T83813 D0U7BH 9815618 EC50 = 25.12 nM T83813 D0U7UD 10826147 Ki = 79 nM T83813 D0U9HE 3693566 Ki = 0.6 nM T83813 D0UZ4J 6604926 Ki = 1200 nM T83813 D0V5HV 4296 IC50 = 150 nM T83813 D0W6RV 10130594 EC50 = 8 nM T83813 D0W8EB 44404905 Ki = 84 nM T83813 D0X6MT 4106 EC50 = 0.38 nM T83813 D0X8LG 11243002 IC50 > 10000 nM T83813 D0XX2U 16006606 Ki = 556 nM T83813 D0XX7J 44451369 Ki = 20 nM T83813 D0Y0SA 135399666 Ki = 34 nM T83813 D0Y9TL 13702393 Ki = 658 nM T83813 D0ZZ4Z 21854226 Ki = 275 nM T25265 D00EQL 66558664 Ki = 2.5 nM T25265 D05FIJ 68210102 Ki = 0.5 nM T25265 D0B4TX 118616529 Ki = 0.15 nM T25265 D0FC9J 118580509 Ki = 0.15 nM T25265 D0LR5O 118580510 Ki = 0.13 nM T25265 CZ92QK 8243546 IC50 > 150000 nM T25265 CH07IQ 9269197 Ki = 700 nM T25265 C24XKI 16348927 IC50 > 200000 nM T25265 CING13 17397370 IC50 > 140000 nM T25265 C7E4KN 17472947 IC50 = 3400 nM T25265 CTZ9J5 17533177 IC50 = 51000 nM T25265 C1M4WO 41507217 IC50 = 2300 nM T25265 C4UDP1 41675187 IC50 > 80000 nM T25265 C73TLV 41676890 IC50 = 57000 nM T25265 CTG1H0 53492732 IC50 < 10 nM T25265 CPL71I 54596764 IC50 = 79 nM T25265 C0DVS4 56597295 IC50 = 3100 nM T25265 CCN65L 56597868 IC50 = 1600 nM T25265 C2FN5Y 57344336 IC50 = 450 nM T25265 CRN54X 57344338 IC50 = 3400 nM T25265 C1WYO9 57344765 IC50 = 29000 nM T25265 CM9VU4 57344770 IC50 = 48000 nM T25265 CPX32V 57345067 IC50 = 48000 nM T25265 C0NO6W 57345068 IC50 = 33000 nM T25265 CYA38P 57345071 IC50 = 59000 nM T25265 CDE9J5 57345180 IC50 = 61000 nM T25265 CUKT25 60160559 IC50 = 400 nM T25265 C2OE4Y 66551041 IC50 = 3100 nM T25265 CFXW24 66575762 EC50 = 500 nM T25265 C3AGQ2 66575763 IC50 = 30 nM T25265 CE7F8K 66575838 EC50 = 300 nM T25265 C2WHT5 66576079 IC50 = 500 nM T25265 C8CQ9D 66576160 IC50 = 1700 nM T25265 CRHX17 66576313 IC50 = 10 nM T25265 CUB4E8 66576790 IC50 = 10 nM T25265 C4Z1RG 67465326 IC50 = 35 nM T25265 CER5F1 67466175 IC50 = 324 nM T25265 C9UH4W 67678991 IC50 > 80000 nM T25265 CS1IO3 67679164 IC50 > 80000 nM T25265 C0ELJ2 67679184 IC50 = 4000 nM T25265 CXV82B 67679189 IC50 > 80000 nM T25265 C5UTO3 67679280 IC50 = 930 nM T25265 CMJ4Y5 67679336 IC50 = 7900 nM T25265 CD0RP6 67679337 IC50 = 3600 nM T25265 C75UVF 67679385 IC50 = 871 nM T25265 C6E4QK 67679426 IC50 > 80000 nM T25265 CP2IF0 67679430 IC50 = 140 nM T25265 CWHJ29 67679449 IC50 = 840 nM T25265 C21SME 67679501 IC50 > 80000 nM T25265 C57OLQ 67679512 IC50 = 51000 nM T25265 CHF74C 67679630 IC50 = 81 nM T25265 CH5L7U 67679638 IC50 > 80000 nM T25265 CKN86F 67679642 IC50 > 80000 nM T25265 C4YC7U 67679664 IC50 = 140 nM T25265 C5QE6A 67988955 IC50 > 50000 nM T25265 C9TP7A 68295073 IC50 = 200 nM T25265 C37VPX 68295468 IC50 = 300 nM T25265 CQN04R 68350784 IC50 = 2400 nM T25265 C60IOE 68350990 IC50 = 5000 nM T25265 CPOR32 68351101 IC50 = 1100 nM T25265 C85YST 68351147 IC50 = 39000 nM T25265 C9N0XY 69671678 IC50 = 24 nM T25265 CU4Y3G 69671822 IC50 > 80000 nM T25265 CG7S0E 69671839 IC50 = 172 nM T25265 CAE7W9 69672405 IC50 > 80000 nM T25265 C6ABM0 69672489 IC50 = 66000 nM T25265 CLA84B 69672582 IC50 = 190 nM T25265 CMI42Q 70872412 EC50 = 700 nM T25265 CC8P3L 70913065 IC50 = 5700 nM T25265 CR85YC 70913076 IC50 = 10 nM T25265 C42TSE 70913205 IC50 = 200 nM T25265 C1CGK3 70913211 IC50 = 100 nM T25265 CXI3A8 70913266 IC50 = 2700 nM T25265 C7E4VI 70913282 IC50 = 200 nM T25265 CFP16O 70913543 IC50 = 20 nM T25265 C0OUV6 71452307 IC50 = 1995 nM T25265 CJ3GP6 71455835 IC50 = 2510 nM T25265 CZ9CS3 71555929 IC50 = 189 nM T25265 CJ0I3E 71715924 IC50 = 118 nM T25265 C1I0YT 78319360 IC50 = 8100 nM T25265 C82LTR 78319363 IC50 = 350 nM T25265 CT2A5Q 78319867 IC50 = 130 nM T25265 CR7T3P 86292233 IC50 = 13 nM T25265 CC5N6Q 86343378 IC50 = 25 nM T25265 CO35HB 86345388 IC50 = 63 nM T25265 CQP15R 86345389 IC50 = 32 nM T25265 C4JO8U 86703409 IC50 = 900 nM T25265 CBQ5C0 86703412 IC50 = 200 nM T25265 CTIB42 86703414 IC50 = 80 nM T25265 CEYR12 86703416 IC50 = 700 nM T25265 CAD5L9 86723730 Ki = 0.7 nM T25265 CYMJ03 86723755 IC50 = 160 nM T25265 C0PD5I 86723793 IC50 = 650 nM T25265 CUY1D4 89584913 IC50 = 1800 nM T25265 CAW4S0 89905749 IC50 = 1400 nM T25265 CNL8E4 90151058 IC50 = 3000 nM T25265 CJDR94 90151131 IC50 = 30 nM T25265 C3YW5E 90151485 IC50 = 100 nM T25265 C1V2IA 90151560 IC50 = 900 nM T25265 CBOC40 90151573 IC50 = 3300 nM T25265 C76SGE 90233370 IC50 = 150 nM T25265 C2RQY7 90233931 IC50 = 5.6 nM T25265 CL3VJ5 90234073 IC50 = 18 nM T25265 C2AI8Q 90234196 IC50 = 28 nM T25265 CPTX74 90234713 IC50 = 56 nM T25265 C37SDG 90246162 IC50 = 41 nM T25265 C43ZSB 90655830 IC50 = 19000 nM T25265 CZEY46 90655831 IC50 = 15000 nM T25265 C5CHN6 90655832 IC50 = 37000 nM T25265 CX60SI 90655833 IC50 > 80000 nM T25265 C63WRS 90655834 IC50 = 1000 nM T25265 C3Q1TF 90655835 IC50 = 920 nM T25265 CITA13 90655836 IC50 = 500 nM T25265 C8HIQ2 90655837 IC50 = 320 nM T25265 CZ0RS5 90655838 IC50 = 1000 nM T25265 CDB7R8 90655839 IC50 = 4900 nM T25265 CMZ7X0 90655840 IC50 > 80000 nM T25265 C3IJL8 90655841 IC50 = 2100 nM T25265 CZV6A3 117778861 IC50 = 1760 nM T25265 CG7LB1 118046535 IC50 = 5700 nM T25265 CO9B4K 118324433 IC50 = 2000 nM T25265 CEZ0I9 118324503 IC50 > 150000 nM T25265 C90NJU 118324514 IC50 = 1300 nM T25265 CL1N2H 118334593 IC50 = 7200 nM T25265 CAKZ31 118572003 Ki = 10 nM T25265 C9CM8K 118572010 Ki = 0.24 nM T25265 C6LAC9 118572014 Ki = 8 nM T25265 CG1M9D 118572015 Ki = 8 nM T25265 CV1F0S 118572016 Ki = 0.25 nM T25265 CA70IU 118572017 Ki = 16 nM T25265 C78LNX 118572065 Ki < 0.1 nM T25265 CCDL26 118572084 Ki = 1260 nM T25265 CIT6E3 118580441 Ki = 0.38 nM T25265 C3AP8U 118580459 Ki = 17 nM T25265 C1OD5P 118580460 Ki = 260 nM T25265 C8PHT6 118580461 Ki = 4.6 nM T25265 CP1U0H 118580466 Ki = 130 nM T25265 CBM9I3 118580471 Ki = 0.15 nM T25265 CQBR41 118580475 Ki = 110 nM T25265 CL8OI0 118580476 Ki = 34 nM T25265 C2KU5S 118580478 Ki = 0.1 nM T25265 CJ72VC 118580479 Ki = 24 nM T25265 CTIA96 118580480 Ki = 135 nM T25265 C8VC0K 118580512 Ki = 0.35 nM T25265 CX8K4L 118580515 Ki < 0.1 nM T25265 C2G6RY 118580520 Ki < 0.1 nM T25265 C5C4KJ 118580531 Ki = 0.22 nM T25265 CD3V9E 118580532 Ki = 0.64 nM T25265 CM5S0F 118580533 Ki = 2.9 nM T25265 C07WGF 118580534 Ki = 0.6 nM T25265 CAB74D 118607629 IC50 = 16 nM T25265 CW6P9U 118616552 IC50 = 6000 nM T25265 CVB79M 118726584 IC50 = 24000 nM T25265 C73TGR 118726585 IC50 = 19000 nM T25265 CX1MY0 118726586 IC50 = 60000 nM T25265 C2JR9D 118726587 IC50 = 120000 nM T25265 CO9K5V 118726588 IC50 = 40000 nM T25265 CZS7A1 118726589 IC50 = 50000 nM T25265 C1DJ0R 118726592 IC50 = 24000 nM T25265 COR67C 118726593 IC50 = 28000 nM T25265 CT83FL 118726594 IC50 = 600 nM T25265 CSO08G 118726595 IC50 = 50000 nM T25265 CIG40B 118726596 IC50 = 2800 nM T25265 CLA1D4 118726597 IC50 = 40000 nM T25265 C5UT7B 118726598 IC50 = 1000 nM T25265 C0JP4I 118726599 IC50 = 3600 nM T25265 CR0JV5 118726600 IC50 = 40000 nM T25265 C8OS9X 122186508 IC50 = 159 nM T25265 C7G8HT 122186509 IC50 = 703 nM T25265 CW34IZ 124175721 IC50 <= 10 nM T25265 COAP71 127025418 IC50 = 14000 nM T25265 CUE2K3 127025970 IC50 > 50000 nM T25265 C4W9MU 127025972 IC50 = 50 nM T25265 CHTY97 127025973 IC50 = 50 nM T25265 C3QOM7 127025974 IC50 = 2200 nM T25265 CS8T2W 127026246 IC50 > 50000 nM T25265 CE13VT 127026272 IC50 = 22000 nM T25265 CW18IG 127026273 IC50 > 50000 nM T25265 C9F4QC 127028788 IC50 = 200 nM T25265 C6B5AP 127029090 IC50 = 18000 nM T25265 C5E9GC 127029640 IC50 > 50000 nM T25265 CS6L3T 127029641 IC50 = 6000 nM T25265 CGA81V 133081962 IC50 = 55 nM T25265 CHC21T 134131668 IC50 = 98 nM T25265 CFO14J 134132569 IC50 = 51 nM T25265 CKN23I 134133285 IC50 = 11 nM T25265 CB4LV2 134134122 IC50 = 375 nM T25265 CH60WZ 134134412 IC50 = 571 nM T25265 CXI6A2 134134567 IC50 = 378 nM T25265 CCRF30 134134857 IC50 = 4140 nM T25265 C19OZF 134135375 IC50 = 88 nM T25265 C54HDM 134135389 IC50 = 17 nM T25265 CTE31R 134137113 IC50 = 975 nM T25265 CO52FX 134137743 IC50 = 185 nM T25265 CYQ7M8 134138451 Ki = 2 nM T25265 CG2NF3 134138932 IC50 = 15700 nM T25265 CJ0L2E 134139550 IC50 = 24 nM T25265 CT2J1B 134142243 IC50 = 17 nM T25265 C47UNK 134143634 IC50 = 237 nM T25265 C1FTQ4 134148232 IC50 = 110 nM T25265 CW25SI 134152139 IC50 = 26800 nM T25265 C64GQS 134152472 IC50 = 44000 nM T25265 CO1IU3 135418643 IC50 = 10300 nM T25265 CRYU96 135463745 IC50 = 22600 nM T25265 CR9LW6 137635406 Ki = 1.5 nM T25265 COZY21 137650028 Ki = 1500 nM T25265 CL9SD7 137652111 Ki = 0.7 nM T25265 C2Y3KW 139211326 IC50 = 12 nM T25265 CCB53A 145960363 IC50 <= 10 nM T25265 C2NIO5 145960476 IC50 <= 10 nM T25265 CR1OQ8 145961928 IC50 <= 10 nM T25265 CO5E2M 145961989 IC50 <= 10 nM T25265 CM5VO6 145962892 IC50 <= 10 nM T25265 CAJ94H 155538504 IC50 > 5000 nM T25265 C75ENB 155538833 IC50 = 328 nM T25265 CPY0B1 155540279 IC50 > 5000 nM T25265 CQ8EU9 155540351 IC50 = 73 nM T25265 C3SLV6 155541578 IC50 > 5000 nM T25265 CJ3SF0 155542049 IC50 = 64 nM T25265 CYPH45 155542586 IC50 = 384 nM T25265 CF3IE0 155542683 IC50 < 10 nM T25265 C9TWY6 155542713 IC50 = 57 nM T25265 C1P6ZK 155542893 IC50 = 540 nM T25265 C7V0NB 155544716 IC50 = 1111 nM T25265 C8I2CL 155545225 IC50 = 25 nM T25265 CWB86N 155546955 IC50 = 32 nM T25265 C2OHG1 155546957 IC50 = 32 nM T25265 C2DY0H 155547180 IC50 = 42 nM T25265 CFJK12 155547766 IC50 = 117 nM T25265 CXVM95 155547840 IC50 = 41 nM T25265 C3GZP6 155547915 IC50 = 26 nM T25265 CY2RI3 155548857 IC50 > 5000 nM T25265 CBW5H1 155548936 IC50 > 2500 nM T25265 CTG91O 155549667 IC50 < 10 nM T25265 C5W6GC 155550181 IC50 = 190 nM T25265 CBA42L 155550828 IC50 > 10000 nM T25265 COAX09 155550957 IC50 = 1016 nM T25265 CM0N8B 155550993 IC50 > 10000 nM T25265 CH50KG 155551023 IC50 = 24 nM T25265 C8TZ2H 155552001 IC50 > 10000 nM T25265 CA95GN 155552788 IC50 = 12 nM T25265 CF8H7X 155553332 IC50 < 10 nM T25265 CWE04H 155554866 IC50 < 10 nM T25265 CE6NL4 155555991 IC50 = 48 nM T25265 CN6WA2 155556614 IC50 < 10 nM T25265 C5SBY9 155557240 IC50 < 10 nM T25265 C5C6GK 155557835 IC50 < 10 nM T25265 C8N2FZ 155557917 IC50 < 10 nM T25265 CHR6N8 155558797 IC50 = 697 nM T25265 C74JAU 155559342 IC50 > 10000 nM T25265 C1XA8H 155560365 IC50 < 10 nM T25265 CJO5K6 155560444 IC50 = 149 nM T25265 CWK90R 155560721 IC50 = 11 nM T25265 C8IX9W 155560875 IC50 = 66 nM T25265 C8K0IE 155561239 IC50 > 2300 nM T25265 COT94K 155563932 IC50 = 17 nM T25265 CPA5R9 155564424 IC50 = 280 nM T25265 C2CAX7 155564971 IC50 > 1250 nM T25265 C18OAD 155567358 IC50 > 5000 nM T25265 CKXG20 155568357 IC50 > 10000 nM T25265 CEIC47 155568678 IC50 > 10000 nM T25265 CW52CQ 155568924 IC50 = 22 nM T25265 CJI41G 155569031 IC50 > 10000 nM T25265 D02TVQ 71268957 IC50 = 174 nM T25265 D09CLP 439155 IC50 = 1900 nM T15497 D06FEA 5280360 EC50 = 3.7 nM T15497 D0WL5V 9867642 Ki = 1160 nM T15497 D00HTY 5280363 IC50 = 380 nM T15497 D00IQH 11677589 Ki > 5000 nM T15497 D00MZK 9911469 Ki = 9600 nM T15497 D00SOZ 44230999 IC50 > 10000 nM T15497 D01SHJ 56944705 IC50 > 10000 nM T15497 D0G6EI 9890801 Ki > 2800 nM T15497 D0M4TJ 44219292 Ki = 9600 nM T15497 D0SP5V 49843471 IC50 > 25000 nM T15497 D0Y3LL 18376177 Ki > 3200 nM T15497 D0W2OT 5311035 Ki > 10000 nM T15497 D02RUO 9807448 Ki > 10000 nM T15497 D08QHS 11296282 IC50 > 20000 nM T15497 C62MKI 1000070 Ki = 63.1 nM T15497 CW59RC 1009982 Ki = 25.12 nM T15497 CAZT67 1283333 Ki = 10 nM T15497 CJ5Q1H 1496731 IC50 = 320 nM T15497 COYI02 1496733 IC50 = 3000 nM T15497 CANV86 1498200 IC50 = 1000 nM T15497 C4GE6B 1498267 IC50 = 430 nM T15497 C52CPY 1498274 IC50 = 580 nM T15497 C3LM8E 1498314 IC50 = 180 nM T15497 CLG45C 1498318 IC50 = 320 nM T15497 C2KC7I 1812712 Ki = 588.84 nM T15497 CLM8P6 2114670 Ki > 25000 nM T15497 C3DXW5 2176335 Ki = 12.88 nM T15497 CU24RF 2285792 Ki < 1122.02 nM T15497 CD2G7Q 2288900 IC50 = 7.943 nM T15497 C4KV3Y 2467304 Ki = 1348.96 nM T15497 C0C5KI 2897583 Ki = 169.82 nM T15497 C3MYH9 3142636 Ki < 1584.89 nM T15497 CE7O8C 3508209 IC50 = 251.19 nM T15497 CQK93L 3686645 Ki = 741.31 nM T15497 CHY95Q 3688070 Ki = 1288.25 nM T15497 CG26SN 3689365 Ki = 61.66 nM T15497 CF32ZT 3717437 Ki < 3801.89 nM T15497 C70STR 3778726 Ki = 34.67 nM T15497 CCWE58 3813994 Ki = 30.9 nM T15497 CLWG42 3855927 Ki = 38.9 nM T15497 C23OQY 5114179 Ki < 1584.89 nM T15497 C2XLU7 5311228 Ki = 1300 nM T15497 CK16QC 5311234 IC50 = 38 nM T15497 CO7N1Z 5311239 EC50 > 10000 nM T15497 CZ15QS 6441607 EC50 = 300 nM T15497 CZA41R 9808508 Ki = 57 nM T15497 C6TA3N 9809136 Ki = 10 nM T15497 CV24TI 9817292 Ki > 100000 nM T15497 CF6Y2K 9820333 IC50 > 3200 nM T15497 CYNX09 9825293 EC50 > 20000 nM T15497 C5J8WP 9830442 Ki = 120 nM T15497 CG3IS9 9830839 Ki > 10000 nM T15497 C9IV7J 9844175 Ki = 4.266 nM T15497 C97MIQ 9865111 Ki = 23000 nM T15497 C5O0RC 9866503 Ki = 28.84 nM T15497 C8J1XO 9868012 Ki = 0.3 nM T15497 C6V1BA 9872741 Ki = 220 nM T15497 CA2I4Z 9873528 Ki = 150 nM T15497 CKMW12 9874010 Ki = 17 nM T15497 CF0HC5 9888589 IC50 > 10000 nM T15497 CFC8G4 9894720 Ki > 3000 nM T15497 CA5N0K 9895436 Ki = 18 nM T15497 CQ0X9R 9909510 IC50 = 3100 nM T15497 CUF02C 9910826 Ki = 15 nM T15497 C7MA6V 9916766 Ki = 200 nM T15497 CN2UX4 9938625 Ki = 47 nM T15497 CICE70 9938626 Ki = 16 nM T15497 C1KAC5 9938669 Ki = 140 nM T15497 C6DQ3W 9938995 Ki = 100 nM T15497 CWDT69 9939791 Ki = 12 nM T15497 CWS81C 9944231 Ki = 34000 nM T15497 C4Q7RI 9953337 Ki = 8500 nM T15497 C3LX4J 9953978 Ki = 3 nM T15497 C6SGH7 9954562 Ki = 9600 nM T15497 C4UK2Q 9955802 Ki = 2500 nM T15497 CVYB74 9956808 IC50 = 6.31 nM T15497 C6ZM4U 9959673 Ki = 770 nM T15497 CCD30P 9960839 Ki = 400 nM T15497 C4Z7BL 9965922 Ki = 68000 nM T15497 C5AF0B 9975502 Ki = 10000 nM T15497 CA85XM 9980905 IC50 = 15.85 nM T15497 CSZ73B 9983512 IC50 = 3.981 nM T15497 CV9Z6B 10000919 IC50 = 63.1 nM T15497 CZUJ52 10001608 IC50 = 10000 nM T15497 C3CMJ9 10003006 IC50 = 5.012 nM T15497 CCD24K 10007859 Ki = 0.1 nM T15497 C8BP6X 10028117 IC50 = 3.981 nM T15497 C2SH9C 10028359 IC50 = 6.31 nM T15497 CR2Q3Z 10030627 IC50 = 2.512 nM T15497 C4SON9 10046844 Ki = 3.548 nM T15497 CQ3GW6 10047541 IC50 = 1100 nM T15497 CVL6T7 10051605 IC50 = 1 nM T15497 CI52XJ 10051678 IC50 = 1.995 nM T15497 CZ6J5T 10051975 IC50 = 50.12 nM T15497 C8HT9A 10052747 IC50 = 5.012 nM T15497 CNE21V 10095268 Ki = 1 nM T15497 CXSF75 10099424 IC50 = 0.631 nM T15497 C6UI2Z 10111602 Ki > 20000 nM T15497 CBYV78 10112486 Ki = 27000 nM T15497 C26QRM 10118889 Ki = 820 nM T15497 C98DZA 10127780 IC50 = 79.43 nM T15497 CS9R6Z 10127791 IC50 = 19.95 nM T15497 C1QI8X 10128061 IC50 = 12.59 nM T15497 C6BOW4 10144273 Ki = 49000 nM T15497 CWN91Y 10150770 IC50 = 100 nM T15497 C9PT3S 10150866 IC50 = 158.49 nM T15497 CCPI72 10151282 IC50 = 31.62 nM T15497 C46EOS 10151840 IC50 = 3.162 nM T15497 C28CIN 10152107 IC50 = 15.85 nM T15497 CG4YV6 10157810 Ki = 151350 nM T15497 C6W9IC 10158725 Ki = 17800 nM T15497 CM3SE6 10168694 Ki = 13000 nM T15497 C6Y3CX 10173065 IC50 = 25.12 nM T15497 C3FXN2 10174660 IC50 = 100 nM T15497 C71GVU 10178073 Ki = 12000 nM T15497 CEM21G 10181606 Ki = 8100 nM T15497 CU47VL 10194556 IC50 = 63.1 nM T15497 C2MEG8 10195119 IC50 = 12.59 nM T15497 CZKM14 10195696 IC50 = 5.012 nM T15497 C6X5CP 10202765 Ki > 100000 nM T15497 CF1NB3 10207799 Ki = 3 nM T15497 C4Y9RW 10215735 IC50 = 6.31 nM T15497 CNRP47 10216080 IC50 = 100 nM T15497 CRA06V 10216528 IC50 = 50.12 nM T15497 CW13VB 10216958 IC50 = 79.43 nM T15497 CP8KN7 10227492 Ki = 1100 nM T15497 C6FM0Z 10238855 IC50 = 39.81 nM T15497 C0ED9Y 10251023 IC50 = 912 nM T15497 CU4RF9 10253022 IC50 = 1.995 nM T15497 C89CXB 10271490 Ki > 10000 nM T15497 CV7H2E 10275911 IC50 > 3200 nM T15497 CL7YG3 10287121 Ki > 13000 nM T15497 CP6D2N 10288374 IC50 = 15.85 nM T15497 C40QFO 10291963 Ki > 100000 nM T15497 CV9QL7 10302378 Ki = 3200 nM T15497 CL65HU 10310187 IC50 = 39.81 nM T15497 CH3W5G 10310313 IC50 = 39.81 nM T15497 CRM34S 10311325 IC50 = 2.512 nM T15497 CXKD46 10322359 IC50 = 2.512 nM T15497 C4JT8F 10324022 IC50 = 0.7943 nM T15497 CE1F7M 10345568 IC50 = 2.512 nM T15497 C58PMI 10345789 IC50 = 1.259 nM T15497 COE09C 10346309 IC50 = 1.259 nM T15497 CPVB42 10347276 IC50 = 5.012 nM T15497 CV8CZ6 10362377 IC50 = 19.95 nM T15497 CB9C1K 10369424 IC50 = 316.23 nM T15497 C51JIX 10389527 IC50 > 10000 nM T15497 CTRJ98 10390894 IC50 = 5.012 nM T15497 CB19MW 10402929 Ki = 63000 nM T15497 CP2GQ0 10411538 IC50 = 3.981 nM T15497 C40XLI 10413628 IC50 = 10 nM T15497 CU6X2V 10454544 IC50 = 10 nM T15497 C8EJL0 10456789 IC50 = 1.259 nM T15497 C59LNJ 10458324 IC50 = 3.162 nM T15497 CLOI24 10459580 IC50 = 0.3981 nM T15497 C2XVE5 10480281 IC50 = 3.162 nM T15497 C3AM2H 10481653 IC50 = 1.585 nM T15497 CI5HA0 10648334 IC50 = 2700 nM T15497 C9YQG5 10670992 IC50 > 10000 nM T15497 C7GY6X 10739351 IC50 = 5000 nM T15497 CY8IB2 10740699 IC50 > 10000 nM T15497 C12SBH 10741017 IC50 = 4600 nM T15497 CG17HE 10741197 IC50 = 364 nM T15497 CKST02 11122314 IC50 > 10000 nM T15497 CL19HV 11154379 IC50 = 79.43 nM T15497 CEI08Z 11155228 Ki = 6700 nM T15497 CC8PQ2 11156167 Ki = 1332 nM T15497 C84HPY 11178058 Ki = 8.71 nM T15497 C9ZVD5 11178059 IC50 = 3.162 nM T15497 C3RDA6 11189804 IC50 = 0.5248 nM T15497 CF6EO3 11210487 Ki = 45000 nM T15497 CE0WA5 11211840 Ki = 0.5888 nM T15497 CG53MW 11213683 IC50 = 15.85 nM T15497 C36UKQ 11223916 IC50 < 1000 nM T15497 CS69HE 11224226 IC50 = 25.12 nM T15497 C9FQC7 11224723 IC50 = 5.012 nM T15497 CA71OC 11235004 IC50 = 6.457 nM T15497 C9WY6K 11235389 Ki = 6.607 nM T15497 C4S5MX 11249458 Ki > 10000 nM T15497 COQJ63 11257814 Ki = 8.318 nM T15497 CU76OJ 11258250 IC50 = 5.012 nM T15497 C70ESM 11269563 Ki > 9000 nM T15497 CI0E7P 11269978 IC50 = 125.89 nM T15497 CSD5K1 11271578 IC50 = 17.78 nM T15497 CC3DK8 11281168 IC50 = 79.43 nM T15497 CWT2X3 11281276 Ki = 20.42 nM T15497 CQFL37 11281855 Ki = 69.18 nM T15497 COS4C2 11294085 Ki = 1080 nM T15497 C9E4SW 11294166 Ki > 20000 nM T15497 CBX1O3 11294771 IC50 = 199.53 nM T15497 C4TIA3 11305124 IC50 = 114.82 nM T15497 CTIR80 11317344 IC50 = 194.98 nM T15497 CFDA92 11326896 IC50 > 3200 nM T15497 CIM8K7 11328569 Ki > 10000 nM T15497 CQ7Z5B 11339406 IC50 > 3200 nM T15497 C3G2ZR 11339792 Ki = 338.84 nM T15497 CG9A1P 11340370 IC50 = 0.1318 nM T15497 C4MC6D 11350546 Ki = 28.18 nM T15497 CBP71Y 11362836 Ki = 431 nM T15497 C3SLX0 11372607 IC50 = 9.772 nM T15497 C4LJ3B 11374485 Ki = 8 nM T15497 C4QD0T 11383800 Ki = 1.122 nM T15497 CKO16T 11384586 IC50 = 7.413 nM T15497 CN2TG7 11387144 Ki > 3000 nM T15497 CN5VD7 11398071 IC50 = 100 nM T15497 C3YS6M 11406237 Ki = 7.943 nM T15497 CTX07D 11407950 IC50 = 14.79 nM T15497 CXPO04 11408533 Ki > 20000 nM T15497 CJ61LG 11418874 Ki = 0.5495 nM T15497 C32EKI 11429983 IC50 = 398.11 nM T15497 CIDT15 11464169 IC50 = 79.43 nM T15497 CZ4K0P 11476788 Ki = 142 nM T15497 C0YZI4 11476911 IC50 = 35.48 nM T15497 CM6Z1E 11486771 IC50 > 3200 nM T15497 CE2JA4 11488860 Ki = 4590 nM T15497 CW3YO5 11494768 IC50 > 25000 nM T15497 CQ6IU7 11509269 IC50 > 10000 nM T15497 CS2LR0 11516353 IC50 > 25000 nM T15497 CF2OM8 11539410 IC50 > 25000 nM T15497 CM7HK0 11551847 IC50 > 25000 nM T15497 CAC6R8 11559437 IC50 = 158.49 nM T15497 CJ2OE0 11575201 IC50 > 20000 nM T15497 C1W2ZK 11577792 Ki > 6000 nM T15497 CS4KE5 11595316 IC50 = 39.81 nM T15497 C7Y6XJ 11597294 Ki = 4400 nM T15497 C2M8HZ 11610353 IC50 > 25000 nM T15497 CGS72I 11618662 IC50 > 20000 nM T15497 C9L5VD 11631813 IC50 > 25000 nM T15497 CD7R5P 11631965 IC50 > 25000 nM T15497 CF7X3A 11640317 Ki = 0.7079 nM T15497 CMB6F9 11653874 IC50 > 25000 nM T15497 CAL96X 11683088 IC50 > 20000 nM T15497 CW8RY9 11689895 IC50 > 25000 nM T15497 C9CM2R 11695689 IC50 > 10000 nM T15497 C3BSV4 11696697 Ki > 13000 nM T15497 CNYK74 11743212 Ki = 48000 nM T15497 CO5CF7 11750434 Ki = 15.49 nM T15497 C8KS5P 11754541 IC50 = 10 nM T15497 C0F8DT 11755633 IC50 = 3.981 nM T15497 CK2EZ6 11962967 Ki = 50.12 nM T15497 CH26TZ 11963255 Ki = 15.85 nM T15497 CR82PA 12112238 Ki = 72000 nM T15497 CX0M2W 12112239 Ki = 5800 nM T15497 C32GBT 12137443 Ki = 18000 nM T15497 CT34LO 13230981 Ki > 13000 nM T15497 CO19GA 14372497 Ki > 7000 nM T15497 C06OGJ 15486805 IC50 = 713 nM T15497 C0L3VU 15486806 IC50 = 1100 nM T15497 CU5J6N 15491229 Ki = 360 nM T15497 CMG0Z1 15491230 Ki = 51000 nM T15497 CWQ8B9 15551228 Ki > 100000 nM T15497 CZ87CN 15907747 Ki = 50 nM T15497 CVEO28 15907748 Ki = 140 nM T15497 CIS83K 15947857 Ki > 9000 nM T15497 C3L0RK 15948325 Ki > 7000 nM T15497 CI61TE 16678098 IC50 > 10000 nM T15497 CS8M2G 18973764 Ki = 230 nM T15497 C6AU1N 21112865 IC50 = 10 nM T15497 CTSG57 21112869 IC50 = 1.995 nM T15497 C13HXO 21112870 IC50 = 6.31 nM T15497 CX08BC 21198692 Ki > 100000 nM T15497 CR37AJ 21362845 Ki = 41000 nM T15497 C6UT1I 21362849 Ki = 8300 nM T15497 C4IFY8 21362851 Ki = 8300 nM T15497 C9HQN0 21362853 Ki = 9500 nM T15497 C6F8QI 21362863 Ki > 97000 nM T15497 CL5O9E 21362867 Ki = 27000 nM T15497 C58NCB 21362869 Ki > 100000 nM T15497 CHS9L6 21362879 Ki = 17500 nM T15497 CW7R1M 21362893 Ki = 4600 nM T15497 C9HD2W 21362900 Ki = 1700 nM T15497 CSUO46 21362905 Ki = 13000 nM T15497 CJ65SZ 21362910 Ki = 11900 nM T15497 CFV24G 21362912 Ki = 3000 nM T15497 C0UT6R 22008966 Ki = 2600 nM T15497 CJ4M7P 22008967 Ki = 2600 nM T15497 C9TSB7 22009003 Ki = 13000 nM T15497 C8SON3 22009004 Ki = 1500 nM T15497 CAML12 22009006 Ki = 8500 nM T15497 C5DGQ4 22009008 Ki = 1500 nM T15497 C5SJ2H 22009011 Ki = 3000 nM T15497 C3D2LR 22990263 Ki = 10000 nM T15497 CFU52S 23583060 IC50 = 10 nM T15497 CG40WR 23661678 IC50 = 2.512 nM T15497 CRIK75 23662249 IC50 = 100 nM T15497 CP2S4J 23663736 Ki > 10000 nM T15497 CT6GV9 23664664 IC50 = 50.12 nM T15497 CAM2U6 23664959 IC50 = 79.43 nM T15497 CGV3N0 23667784 Ki = 0.3162 nM T15497 C4WEN7 23667788 Ki = 1.995 nM T15497 C7UER5 23667790 Ki = 1.995 nM T15497 CIM16O 23673471 IC50 = 158.49 nM T15497 C71WTB 23674081 IC50 = 25.12 nM T15497 CLTO53 23676882 IC50 = 251.19 nM T15497 CQ6VS5 23677039 IC50 = 100 nM T15497 CU5S0K 23678183 IC50 = 50.12 nM T15497 CSAG29 23678185 IC50 = 25.12 nM T15497 CUA78E 23678186 IC50 = 25.12 nM T15497 CX1R5S 23678188 Ki = 1.585 nM T15497 C1O5LD 23678203 IC50 = 7.943 nM T15497 CV16MQ 23678676 IC50 = 39.81 nM T15497 C5D3RZ 23683143 IC50 = 10 nM T15497 C2F8GY 23684396 IC50 = 630.96 nM T15497 C9H4WT 23686961 Ki = 2.512 nM T15497 CWZF16 23690263 IC50 = 79.43 nM T15497 CKVG18 23690266 IC50 = 39.81 nM T15497 C4PGA6 23690271 IC50 = 19.95 nM T15497 C1HW9I 23690284 IC50 = 199.53 nM T15497 CGPU68 23690392 IC50 = 63.1 nM T15497 CM83CJ 23694419 IC50 = 39.81 nM T15497 C42JWU 23696344 Ki = 0.7943 nM T15497 C26ANU 23696680 IC50 = 12.59 nM T15497 CD78UH 23696969 IC50 = 31.62 nM T15497 CE6JU7 23696971 IC50 = 39.81 nM T15497 CASU54 23696973 Ki = 7.943 nM T15497 C7EV5C 23710225 IC50 = 100 nM T15497 C01OAQ 23710226 IC50 = 100 nM T15497 CZ58NG 23713252 IC50 = 12.59 nM T15497 C42LYP 24765153 Ki = 28500 nM T15497 CF72YI 24765671 Ki >= 785 nM T15497 C31JZP 24765672 Ki >= 2500 nM T15497 C4QX7Y 24765675 Ki >= 930 nM T15497 CL7Z9U 24765768 Ki >= 110 nM T15497 C5A1CB 24783314 IC50 = 316.23 nM T15497 C0R6TW 24784836 Ki = 0.3981 nM T15497 CYD4V9 24784839 IC50 = 100 nM T15497 CV4JQ8 24784840 IC50 = 50.12 nM T15497 C58LYT 24785079 IC50 = 63.1 nM T15497 CM92HY 24785588 IC50 = 25.12 nM T15497 CE61RT 24785591 IC50 = 50.12 nM T15497 C1XML0 24785594 IC50 = 3.981 nM T15497 CHQS54 24785595 IC50 = 63.1 nM T15497 C6A1IF 24785862 IC50 = 794.33 nM T15497 C1XT9F 24894000 IC50 = 100 nM T15497 C5JI2X 24894001 IC50 = 50.12 nM T15497 C5WO6H 24894002 IC50 = 12.59 nM T15497 CFQA40 24952577 Ki > 7282 nM T15497 CD98IN 24952580 Ki > 456 nM T15497 C81WVN 24952927 Ki > 5474 nM T15497 CZT83E 24952928 Ki > 501 nM T15497 C8YHX3 24953283 Ki > 224 nM T15497 CZ93FO 24953285 Ki > 628 nM T15497 C17JTY 24953286 Ki > 2226 nM T15497 CFT0W5 24953624 Ki > 4992 nM T15497 C42VMD 24953625 Ki > 3461 nM T15497 C7B2EW 24953628 Ki > 2117 nM T15497 CNME84 25002355 IC50 = 5.012 nM T15497 CXQJ67 25002382 Ki >= 1291 nM T15497 C5Z0AX 25002703 IC50 = 10 nM T15497 CN5SH9 25003075 Ki = 20000 nM T15497 CI5QA1 25005134 IC50 = 25.12 nM T15497 CT47LQ 25005494 IC50 = 6.31 nM T15497 CIP60C 25005495 IC50 = 7.943 nM T15497 CQ34XS 25005499 IC50 = 5.012 nM T15497 CA1VI6 25007720 IC50 = 10 nM T15497 CH1M3Y 25008273 IC50 < 1000 nM T15497 C2GO4D 28568627 Ki = 25.12 nM T15497 CR10FW 30897313 IC50 > 30000 nM T15497 CNOF71 44138108 Ki = 28500 nM T15497 CSRV98 44157014 IC50 = 1420 nM T15497 C2O0NL 44230575 IC50 > 10000 nM T15497 CR68BA 44250281 Ki > 10000 nM T15497 CN90FE 44269464 Ki > 13000 nM T15497 C1L0ET 44269468 Ki > 13000 nM T15497 C5KRQ4 44269486 Ki > 13000 nM T15497 CL6M2P 44269516 Ki > 13000 nM T15497 CON8R9 44269520 Ki > 13000 nM T15497 C6MBG0 44269521 Ki > 13000 nM T15497 CZ3Q1L 44269523 Ki > 13000 nM T15497 CRL61O 44269532 Ki > 13000 nM T15497 C1Z4LU 44269540 Ki > 13000 nM T15497 CM72FA 44269542 Ki > 13000 nM T15497 CN0JV2 44269543 Ki > 13000 nM T15497 C28UJH 44269544 Ki > 13000 nM T15497 CR1IY6 44269568 Ki > 13000 nM T15497 CI3C9O 44269596 Ki > 13000 nM T15497 CC0EW9 44269597 Ki > 13000 nM T15497 CWJC89 44285146 IC50 = 10000 nM T15497 C5P9CF 44285208 IC50 > 10000 nM T15497 CCD2S1 44285209 IC50 > 10000 nM T15497 C9U7YH 44285251 IC50 > 10000 nM T15497 C6EZ1R 44285252 IC50 > 10000 nM T15497 CS64GQ 44285310 EC50 > 20000 nM T15497 CDP9F2 44285328 IC50 = 3450 nM T15497 CY37TX 44289792 Ki > 100000 nM T15497 C4SEW6 44290266 Ki = 4.5 nM T15497 C4F8YR 44290494 Ki = 50000 nM T15497 CS7RH0 44320126 Ki = 2800 nM T15497 CLR9F5 44320272 Ki = 3700 nM T15497 CKYS39 44320294 Ki = 7500 nM T15497 CH6TK1 44320321 Ki = 1800 nM T15497 CYI1O0 44320373 Ki = 8600 nM T15497 C0V3OA 44320388 Ki = 15000 nM T15497 C01HGT 44320405 Ki = 2800 nM T15497 CS58ZQ 44320433 Ki = 83 nM T15497 C1R5LX 44324302 Ki = 10800 nM T15497 CGV86S 44324309 Ki = 2800 nM T15497 C0K6QY 44324310 Ki = 1200 nM T15497 CS52ZR 44324368 Ki = 21000 nM T15497 CM72WE 44349503 Ki = 2600 nM T15497 C9PO1Q 44349528 Ki = 35000 nM T15497 C1R7HU 44349531 Ki = 9300 nM T15497 CHO7X0 44349551 Ki = 85000 nM T15497 CLN63A 44377464 Ki > 100000 nM T15497 CJIS72 44390782 Ki > 9000 nM T15497 C43VIA 44390806 Ki > 9000 nM T15497 CB8H4V 44390831 Ki = 17000 nM T15497 C0YXP5 44392456 Ki = 4 nM T15497 CXB76Y 44392460 Ki = 6 nM T15497 CN1L7E 44392477 Ki = 260 nM T15497 C1YKS6 44392479 Ki = 52 nM T15497 CP2O4K 44392512 Ki = 23 nM T15497 CI2KP5 44392527 Ki = 9 nM T15497 CWL1X4 44400355 Ki > 1000 nM T15497 C76QVA 44402710 Ki > 1000 nM T15497 CRAX23 44402824 Ki > 1000 nM T15497 CYG6Q2 44409742 IC50 > 3200 nM T15497 CKM6S2 44409910 IC50 = 18550 nM T15497 CS42GV 44409918 IC50 > 3200 nM T15497 CZ59NQ 44410764 Ki < 1000 nM T15497 CI8K5T 44410767 Ki < 1000 nM T15497 C3R0TG 44410777 Ki < 1000 nM T15497 CYCU18 44410874 IC50 = 7.943 nM T15497 C5GP0K 44410930 IC50 < 1000 nM T15497 C2GRC7 44410931 Ki = 52.48 nM T15497 CDX19R 44413003 IC50 = 12.59 nM T15497 CDL3A0 44413013 IC50 = 12.59 nM T15497 CAV5E6 44413014 IC50 = 100 nM T15497 C2JGA9 44413078 IC50 = 25.12 nM T15497 CFH78Y 44413079 IC50 = 100 nM T15497 C90YGL 44413091 IC50 = 79.43 nM T15497 COR3J5 44413092 IC50 = 6.31 nM T15497 CW08LP 44413101 IC50 = 5.012 nM T15497 CO2C4S 44413102 IC50 = 25.12 nM T15497 CVO38X 44413104 IC50 = 6.31 nM T15497 CFBP14 44413109 IC50 = 19.95 nM T15497 C4PJS3 44413110 IC50 = 398.11 nM T15497 CBT5J0 44413120 IC50 = 630.96 nM T15497 C2I5KL 44413122 IC50 = 79.43 nM T15497 C2OT6J 44413123 IC50 = 12.59 nM T15497 C9U6BP 44413124 IC50 = 10 nM T15497 C1NE0R 44413128 IC50 = 15.85 nM T15497 C62ZXT 44413129 IC50 = 10 nM T15497 C9OP2A 44413135 IC50 = 5.012 nM T15497 CO9C3V 44413140 IC50 = 19.95 nM T15497 CIH8Q9 44413141 IC50 = 7.943 nM T15497 CP5UI1 44413152 IC50 = 2.512 nM T15497 CJF2C0 44413153 IC50 = 251.19 nM T15497 CE5U2A 44413163 IC50 = 39.81 nM T15497 CAZ9O8 44413164 IC50 = 50.12 nM T15497 CE3FK7 44413172 IC50 = 50.12 nM T15497 C0PXB6 44413173 IC50 = 25.12 nM T15497 C8TV2W 44413181 IC50 = 39.81 nM T15497 CL59OU 44413188 IC50 = 3.981 nM T15497 CS1ET9 44413189 IC50 < 1000 nM T15497 COZN14 44413197 IC50 = 794.33 nM T15497 C7UX3Y 44413198 IC50 < 1000 nM T15497 CZ9YK6 44413199 IC50 = 199.53 nM T15497 COI65W 44413200 IC50 = 39.81 nM T15497 C0J3HC 44413205 IC50 = 125.89 nM T15497 CUF34D 44413206 IC50 = 39.81 nM T15497 CH6J7L 44413218 IC50 = 31.62 nM T15497 CL07GR 44413360 IC50 = 100 nM T15497 C1J9UC 44413383 IC50 = 15.85 nM T15497 C8WQK7 44415850 IC50 = 676.08 nM T15497 CZY71Q 44415953 Ki < 1995.26 nM T15497 CV0XB7 44415969 Ki = 977.24 nM T15497 CLJV80 44416027 Ki < 1995.26 nM T15497 CQA7Z4 44416047 Ki < 1995.26 nM T15497 CG2LM3 44416096 Ki < 1995.26 nM T15497 CRL17O 44416110 IC50 = 123.03 nM T15497 C5DGF9 44416127 IC50 = 426.58 nM T15497 CW0K5P 44416141 IC50 = 457.09 nM T15497 CLVH03 44416198 IC50 = 309.03 nM T15497 CU1CI7 44416199 Ki = 1122.02 nM T15497 C6DBS9 44416210 IC50 = 575.44 nM T15497 CN50JT 44416211 IC50 = 1230.27 nM T15497 CY67WB 44416229 Ki < 1995.26 nM T15497 CXGF21 44416269 Ki < 1995.26 nM T15497 C4AZ5N 44416283 Ki < 1995.26 nM T15497 CDY3V7 44416284 Ki < 1995.26 nM T15497 C14HGB 44416285 Ki < 1995.26 nM T15497 CIB2W5 44419347 Ki = 6700 nM T15497 CF35LY 44419350 Ki = 23000 nM T15497 CNK1X9 44419351 Ki = 6700 nM T15497 C91JXT 44419374 Ki = 19000 nM T15497 CNF4W2 44419379 Ki = 19000 nM T15497 CS3IW4 44419380 Ki = 2300 nM T15497 CBQ01L 44419384 Ki = 2300 nM T15497 CV8AU4 44426661 IC50 = 1.995 nM T15497 CHBC62 44426662 IC50 = 7.943 nM T15497 CI25WU 44426663 IC50 = 15.85 nM T15497 CJ68LW 44426664 IC50 = 12.59 nM T15497 C5KO3T 44426665 IC50 = 2.512 nM T15497 CSY2T7 44426666 IC50 = 1.995 nM T15497 C7Z6RH 44426667 IC50 = 5.012 nM T15497 CL3DA1 44426668 IC50 = 1.995 nM T15497 CK9WG8 44426669 IC50 = 0.3981 nM T15497 CW0X7Z 44426670 IC50 = 6.31 nM T15497 CV4O9N 44426671 IC50 = 12.59 nM T15497 CP87VW 44426672 IC50 = 5.012 nM T15497 CW7YJ0 44426673 IC50 = 2.512 nM T15497 CGI7Q5 44426674 IC50 = 79.43 nM T15497 C1WK3B 44426675 IC50 = 25.12 nM T15497 C6SB9F 44430672 IC50 = 6.31 nM T15497 C1FR2V 44430673 IC50 = 6.31 nM T15497 CPO1A3 44430674 IC50 = 6.31 nM T15497 CR9C7X 44430675 IC50 = 316.23 nM T15497 C5SM4K 44430676 IC50 = 158.49 nM T15497 C3NIP2 44430677 IC50 = 251.19 nM T15497 C4DGQ8 44430678 IC50 = 125.89 nM T15497 CA6UK1 44430689 IC50 = 3.981 nM T15497 CRX63K 44430690 IC50 = 3.981 nM T15497 CZI19D 44430691 IC50 = 5.012 nM T15497 CSK2L7 44430693 IC50 = 5.012 nM T15497 C5X6HP 44430695 IC50 = 10 nM T15497 C2H8OC 44430697 IC50 = 12.59 nM T15497 CO8QG7 44430698 IC50 = 3.981 nM T15497 CJ41UQ 44430699 IC50 = 3.162 nM T15497 CHO4K6 44430700 IC50 = 0.5012 nM T15497 CU65RE 44430701 IC50 = 3.981 nM T15497 C6XTQ5 44430702 IC50 = 1.995 nM T15497 COA56V 44430703 IC50 = 1.259 nM T15497 CZH6C2 44430704 IC50 = 0.7943 nM T15497 C1DX7G 44430705 IC50 = 1.585 nM T15497 C7OG6H 44430706 IC50 = 1.259 nM T15497 C8MT0H 44430707 IC50 = 1.585 nM T15497 C97PXQ 44430708 IC50 = 1.259 nM T15497 CZ2MO4 44430709 IC50 = 1.995 nM T15497 CBL28M 44430710 IC50 = 1.259 nM T15497 C09ZIS 44430711 IC50 = 5.012 nM T15497 CQ9MS4 44430712 IC50 = 7.943 nM T15497 C01PQW 44430772 IC50 = 398.11 nM T15497 CWG71J 44430773 IC50 = 398.11 nM T15497 C3RGU1 44430774 IC50 = 199.53 nM T15497 CZ4W6P 44430775 IC50 = 1.585 nM T15497 C3HB7E 44430776 IC50 = 39.81 nM T15497 CB1Y4W 44430777 IC50 = 199.53 nM T15497 C4TZH0 44432326 IC50 = 3.981 nM T15497 CTP8N0 44432327 IC50 = 2.512 nM T15497 CCUD37 44432328 IC50 = 79.43 nM T15497 C0RJS3 44432329 IC50 = 7.943 nM T15497 CNPF91 44432330 IC50 = 25.12 nM T15497 CS89TQ 44432331 IC50 < 1000 nM T15497 C6I3WD 44432332 IC50 = 125.89 nM T15497 CXN7W0 44432333 IC50 = 199.53 nM T15497 CP2VW4 44432334 IC50 = 501.19 nM T15497 C32JKO 44432335 IC50 = 19.95 nM T15497 CYM93G 44432336 IC50 = 31.62 nM T15497 C21UQM 44432337 IC50 = 19.95 nM T15497 C38IUP 44432338 IC50 = 7.943 nM T15497 CX2CF3 44432339 IC50 = 3.981 nM T15497 C0YB1L 44432341 IC50 = 15.85 nM T15497 C8Y6HR 44432343 IC50 = 50.12 nM T15497 C7SRQ3 44432344 IC50 = 15.85 nM T15497 CA3I6R 44432346 IC50 = 25.12 nM T15497 CPW8S3 44432348 IC50 = 2.512 nM T15497 C7EB4G 44432350 IC50 = 12.59 nM T15497 CD58ME 44432353 IC50 = 63.1 nM T15497 CMBP27 44432355 IC50 = 5.012 nM T15497 CQ41MO 44432357 IC50 = 501.19 nM T15497 C2MH7I 44432358 IC50 = 63.1 nM T15497 CLN16F 44432359 IC50 = 19.95 nM T15497 C4S7MR 44432360 IC50 = 501.19 nM T15497 CQR15T 44432361 IC50 = 25.12 nM T15497 CK50TQ 44432362 IC50 = 63.1 nM T15497 C37GUZ 44432365 IC50 = 63.1 nM T15497 C1PLI8 44432366 IC50 = 39.81 nM T15497 C06PCM 44432367 IC50 = 1.585 nM T15497 C1IZH5 44432368 IC50 = 630.96 nM T15497 CXPQ51 44432369 IC50 = 25.12 nM T15497 CCT9Y3 44432370 IC50 = 39.81 nM T15497 CFUA74 44432371 IC50 = 39.81 nM T15497 CFA5R4 44432372 IC50 = 125.89 nM T15497 CWU9P3 44432373 IC50 = 251.19 nM T15497 C49EJP 44432374 IC50 = 125.89 nM T15497 C3K7CX 44432375 IC50 = 63.1 nM T15497 C73KVQ 44432376 IC50 = 39.81 nM T15497 CX0QN7 44432377 IC50 = 199.53 nM T15497 C0GT2K 44432378 IC50 = 63.1 nM T15497 CH9Y2D 44432379 IC50 = 63.1 nM T15497 CIR81X 44432380 IC50 = 39.81 nM T15497 CMNQ76 44432381 IC50 = 501.19 nM T15497 CZU89A 44432382 IC50 = 158.49 nM T15497 C8GN3E 44432865 IC50 = 63 nM T15497 CQ28ZM 44432866 Ki = 398.11 nM T15497 C0A3FT 44432868 Ki = 316.23 nM T15497 C4VB8E 44432869 IC50 = 125.89 nM T15497 CK9RG3 44432870 Ki = 39.81 nM T15497 CHC74W 44432872 IC50 = 63.1 nM T15497 C4QFB0 44432875 IC50 = 6.31 nM T15497 CW56NG 44432876 IC50 = 3.981 nM T15497 CXA1B6 44432878 IC50 = 7.943 nM T15497 CQ24PR 44432879 IC50 = 6.31 nM T15497 CVD6R2 44432883 IC50 = 12.59 nM T15497 C3EG1D 44432886 IC50 = 50.12 nM T15497 CWDC28 44432888 IC50 = 199.53 nM T15497 C7TAX1 44432890 IC50 = 501.19 nM T15497 C0CNL8 44432892 IC50 = 316.23 nM T15497 CZQL38 44432896 IC50 = 79.43 nM T15497 CE1TA5 44432905 IC50 = 158.49 nM T15497 CLZC73 44432907 IC50 = 63.1 nM T15497 C7RVL1 44432908 IC50 = 63.1 nM T15497 C3AWX8 44432910 IC50 = 19.95 nM T15497 CW15LG 44432912 Ki = 100 nM T15497 CSM2K0 44432919 IC50 = 31.62 nM T15497 CE6LR8 44432921 IC50 = 39.81 nM T15497 C9O0YW 44432922 IC50 = 7.943 nM T15497 C4YA1N 44432923 IC50 = 25.12 nM T15497 CB8P1N 44432925 IC50 = 501.19 nM T15497 C51NCP 44432926 IC50 = 19.95 nM T15497 CPO02Z 44439583 Ki = 204.17 nM T15497 CGK92F 44439584 Ki = 89.13 nM T15497 C3UB1E 44439585 Ki = 66.07 nM T15497 CZB1E2 44439586 Ki = 3.715 nM T15497 CK0D5R 44439589 Ki = 61.66 nM T15497 C3YNC2 44439590 Ki = 19.05 nM T15497 C97TEH 44439591 Ki = 28.84 nM T15497 CQ4Z6R 44439592 Ki = 31.62 nM T15497 CL1AN7 44439593 Ki = 69.18 nM T15497 CADL90 44439594 Ki = 165.96 nM T15497 CR54CT 44439595 Ki = 169.82 nM T15497 C71JMQ 44439596 Ki = 239.88 nM T15497 C52LSN 44439597 Ki = 707.95 nM T15497 C9BAW7 44439599 Ki = 1659.59 nM T15497 CA48KQ 44439601 Ki = 1995.26 nM T15497 C61JKE 44439602 Ki < 3162.28 nM T15497 C8AHT3 44439606 Ki = 79.43 nM T15497 C0FW8K 44439608 Ki = 426.58 nM T15497 C7B8PQ 44439609 Ki = 251.19 nM T15497 CM2LD5 44439612 Ki = 22.91 nM T15497 CIA82W 44439614 Ki = 208.93 nM T15497 CV2P9Z 44439615 Ki = 134.9 nM T15497 CFM9W8 44439617 Ki = 1071.52 nM T15497 C6A2KM 44439618 Ki < 1000 nM T15497 CY6O9R 44439619 Ki < 1000 nM T15497 C8YV9P 44439620 Ki = 199.53 nM T15497 CY5I3Q 44439621 Ki = 794.33 nM T15497 C5F2RL 44439622 Ki < 1000 nM T15497 C57GIX 44439627 Ki < 1000 nM T15497 C2M0EH 44439628 Ki < 1000 nM T15497 CJ90NV 44439629 Ki = 398.11 nM T15497 CHJ4P3 44439630 Ki = 72.44 nM T15497 CGS0P7 44442327 Ki > 10000 nM T15497 CF32IP 44442331 Ki = 10000 nM T15497 CQFV46 44448347 IC50 = 15.85 nM T15497 COD4S1 44448598 IC50 = 39.81 nM T15497 C65FEA 44448665 IC50 = 6.31 nM T15497 C2QJI5 44448848 IC50 < 1000 nM T15497 CT52VS 44448851 IC50 = 100 nM T15497 CE57UV 44448885 IC50 = 39.81 nM T15497 C2X1MH 44448887 IC50 = 39.81 nM T15497 CE1OX9 44448890 IC50 = 251.19 nM T15497 C0WGH5 44448892 IC50 = 125.89 nM T15497 C1RWF9 44448921 IC50 = 630.96 nM T15497 CIM94R 44448922 IC50 < 1000 nM T15497 CTAR71 44448924 IC50 < 1000 nM T15497 CX85KO 44448928 IC50 = 31.62 nM T15497 C8KQP9 44448929 Ki = 3.981 nM T15497 C5GLI2 44448953 IC50 = 158.49 nM T15497 C3ZLT0 44448954 IC50 = 6.31 nM T15497 C3UV1I 44448955 Ki = 19.95 nM T15497 CIU0C5 44448956 IC50 = 31.62 nM T15497 CZ86ME 44448957 IC50 = 39.81 nM T15497 C69LIW 44448980 IC50 = 50.12 nM T15497 C5POS4 44448983 Ki = 63.1 nM T15497 C7N1IY 44448984 Ki = 1.259 nM T15497 CR31DI 44448985 IC50 < 1000 nM T15497 C94ZPE 44448986 Ki = 0.5 nM T15497 CZ0Y2S 44449009 IC50 = 158.49 nM T15497 CN37ZH 44449011 IC50 = 100 nM T15497 CB7D5P 44449013 IC50 = 6.31 nM T15497 C2FJ1X 44449036 Ki = 1 nM T15497 CYB42T 44449060 IC50 = 10 nM T15497 CSA84U 44449089 Ki = 0.0631 nM T15497 C3E7YJ 44449112 Ki = 0.1995 nM T15497 C6EA2I 44449114 IC50 = 39.81 nM T15497 CS93ME 44449142 IC50 < 1000 nM T15497 CE63YD 44449145 Ki = 12.59 nM T15497 CROB43 44449178 IC50 < 1000 nM T15497 C7N4PH 44449206 IC50 = 1000 nM T15497 CDBE16 44450497 Ki = 2174 nM T15497 CKB9V3 44454965 IC50 = 10 nM T15497 C1NW2S 44455021 IC50 < 1000 nM T15497 C7MDR3 44455091 IC50 = 316.23 nM T15497 C25BPW 44455131 IC50 = 39.81 nM T15497 CUY9J0 44455167 Ki = 15.85 nM T15497 C86HFM 44455203 IC50 = 316.23 nM T15497 C5INZ7 44455243 IC50 = 630.96 nM T15497 CP76KO 44455299 IC50 = 158.49 nM T15497 C8IJC9 44455300 IC50 = 79.43 nM T15497 C78WMD 44455411 IC50 = 794.33 nM T15497 CJ1N7W 44455415 IC50 < 1000 nM T15497 CTF7Y2 44455437 IC50 < 1000 nM T15497 CWVU28 44455440 IC50 = 630.96 nM T15497 CUHD74 44564571 IC50 > 10000 nM T15497 CA05LN 44564804 IC50 = 3860 nM T15497 C6XE0K 44564841 IC50 > 10000 nM T15497 CND54C 44564892 IC50 = 5320 nM T15497 C18GXI 44564937 IC50 > 10000 nM T15497 CZ74GB 44564990 IC50 = 1370 nM T15497 CFC3H9 44568183 IC50 = 6.31 nM T15497 CZR05P 44568186 IC50 = 12.59 nM T15497 C0KY1D 44568188 IC50 = 7.943 nM T15497 CUT2X9 44568217 IC50 = 12.59 nM T15497 CSZ41P 44568302 IC50 = 12.59 nM T15497 CHM78D 44568304 IC50 = 10 nM T15497 C8SLM0 44568506 IC50 = 25.12 nM T15497 C86RTU 44568508 IC50 = 501.19 nM T15497 CS9H7T 44568510 IC50 = 630.96 nM T15497 C02OQZ 44568512 IC50 = 125.89 nM T15497 C31FDP 44568552 IC50 = 501.19 nM T15497 C6EJ1N 44568554 IC50 = 251.19 nM T15497 CXCN75 44568556 IC50 = 12.59 nM T15497 C9BQO0 44568595 IC50 = 100 nM T15497 C86UNJ 44568598 IC50 = 39.81 nM T15497 CQR7D0 44568600 IC50 = 50.12 nM T15497 C5L1DJ 44568630 IC50 = 50.12 nM T15497 CIR6N9 44568632 IC50 = 50.12 nM T15497 COVH20 44568634 IC50 = 100 nM T15497 C1TH4O 44568636 IC50 = 39.81 nM T15497 CT8E2H 44568659 IC50 = 100 nM T15497 CE2RP3 44568661 IC50 = 79.43 nM T15497 C3XDL8 44568663 IC50 = 50.12 nM T15497 COMC91 44568665 IC50 = 31.62 nM T15497 CJAC25 44568703 IC50 = 7.943 nM T15497 CJ8HU1 44568705 IC50 = 7.943 nM T15497 CE2WD3 44568707 IC50 = 5.012 nM T15497 CTGH71 44568709 IC50 = 6.31 nM T15497 C54WIO 44568756 IC50 = 6.31 nM T15497 CVT79H 44568758 IC50 = 7.943 nM T15497 C7ZEI3 44568760 IC50 = 25.12 nM T15497 CN07YJ 44568762 IC50 = 15.85 nM T15497 C07ODW 44570000 IC50 = 6354 nM T15497 CTW6L7 44570712 IC50 = 11600 nM T15497 CGX17U 44571206 IC50 = 6900 nM T15497 CXQI89 44571354 IC50 = 1400 nM T15497 C9D6YH 44581576 IC50 = 316.23 nM T15497 COM89N 44581577 IC50 > 1000 nM T15497 CD1C6F 44581579 IC50 > 1000 nM T15497 C0X9TK 44581618 IC50 > 1000 nM T15497 CD1N3Q 44581620 IC50 = 19.95 nM T15497 C4P5NW 44581621 IC50 = 794.33 nM T15497 C86WXN 44581654 IC50 = 501.19 nM T15497 C29HWE 44581655 IC50 = 79.43 nM T15497 C30CSH 44581656 IC50 = 125.89 nM T15497 CWNX80 44611364 IC50 = 20 nM T15497 C9WJ1O 44611631 IC50 = 60 nM T15497 C6V9JK 44611633 IC50 = 60 nM T15497 CZ2R1S 44611763 IC50 = 30 nM T15497 CI97ZH 44611764 IC50 = 50 nM T15497 C5PT0Z 44626877 IC50 = 8104 nM T15497 CQIK27 44627395 IC50 = 7959 nM T15497 C4W1ZG 44627515 IC50 = 360 nM T15497 C6XVT4 45265995 IC50 < 1000 nM T15497 CJ5Q7H 45265996 IC50 < 1000 nM T15497 C5AY6M 46220498 IC50 = 50 nM T15497 CDH0X5 46220500 IC50 = 2.4 nM T15497 CS4F0X 46879894 IC50 > 20000 nM T15497 C0A2CI 46890616 Ki >= 504 nM T15497 CW52VH 46890658 Ki >= 260 nM T15497 CXQ2W0 46890659 Ki >= 580 nM T15497 CQ20RC 46890660 Ki >= 100 nM T15497 CM63IN 46926351 IC50 = 0.1288 nM T15497 CTR7Q0 49850345 Ki > 50118.72 nM T15497 CM06FG 50898361 Ki > 9500 nM T15497 CF1ZU9 52945294 Ki > 20000 nM T15497 C4K6BH 52946883 Ki > 10000 nM T15497 CWR1Z7 56665984 Ki > 13000 nM T15497 CWY81B 57390334 IC50 > 1000 nM T15497 C1Z2WO 57392102 IC50 = 39.81 nM T15497 C94YAR 57393867 IC50 = 100 nM T15497 CV5Q0L 57393868 IC50 = 25.12 nM T15497 CMY6D0 57393869 IC50 = 10 nM T15497 CR6IN7 57395493 IC50 = 251.19 nM T15497 C0M3VY 57395594 IC50 = 63.1 nM T15497 CDN93B 57395595 IC50 = 63.1 nM T15497 C7YA2U 57397404 IC50 = 19.95 nM T15497 C83LFV 57399015 IC50 = 501.19 nM T15497 CR43XV 57399080 IC50 = 1.995 nM T15497 C6Y1IH 57400734 IC50 = 125.89 nM T15497 CD8WZ9 57402583 IC50 > 1000 nM T15497 CP7A2U 58905349 IC50 > 20000 nM T15497 CB1N8J 58905358 IC50 > 20000 nM T15497 C1CFM4 58905388 IC50 > 20000 nM T15497 CGY68V 59179219 IC50 = 330 nM T15497 CGFQ58 59179237 IC50 = 1000 nM T15497 C54DPL 59179256 IC50 = 80 nM T15497 C0U1HA 59179260 Ki = 8 nM T15497 CO2F1T 59179264 IC50 = 500 nM T15497 C6OWM9 59179265 IC50 = 20 nM T15497 C18BHX 59179268 IC50 = 2 nM T15497 C09BZC 59179280 IC50 = 20 nM T15497 C6MN0U 59179283 IC50 = 120 nM T15497 CF1W5X 59179287 IC50 = 100 nM T15497 C0U4QG 59179305 IC50 = 40 nM T15497 CDV82L 59179306 IC50 > 100 nM T15497 C5MS1I 59179877 IC50 > 100 nM T15497 CZ0DX1 59179878 IC50 = 4 nM T15497 CK7T6D 59179887 Ki = 0.45 nM T15497 C71SJQ 59179893 IC50 = 80 nM T15497 C37YJV 59179904 IC50 = 2 nM T15497 CAH15K 59179908 IC50 = 4.5 nM T15497 C4CIH9 59179917 IC50 = 0.3 nM T15497 C54UTN 59179923 IC50 = 16 nM T15497 CT1Q6H 59179924 IC50 = 4 nM T15497 CIZ0E4 59179928 IC50 = 16 nM T15497 CY5A9T 59179932 IC50 = 120 nM T15497 CTR67N 59179936 IC50 = 1.1 nM T15497 CEG62U 59179944 IC50 = 0.7 nM T15497 C9MXC8 59179967 IC50 = 39 nM T15497 CYU8B1 59179968 IC50 = 80 nM T15497 C58YLU 59179969 IC50 = 30 nM T15497 C6IWV8 59179970 IC50 = 500 nM T15497 C5MTJ9 59179971 IC50 = 12 nM T15497 CV9J7B 59179973 IC50 = 19 nM T15497 C2I1SE 59179974 IC50 = 12 nM T15497 C1YPB7 59179977 IC50 = 32 nM T15497 CCD2K6 59179992 IC50 = 1000 nM T15497 CP3XC1 59180001 IC50 = 100 nM T15497 CB81OX 59180015 IC50 = 200 nM T15497 CVC72I 59554822 Ki = 220 nM T15497 CCXA68 59554824 Ki = 120 nM T15497 CNUA34 66857670 Ki = 89 nM T15497 C1WA3L 66857738 Ki = 149 nM T15497 CU5V8I 66858111 Ki = 802 nM T15497 CF47LN 68258993 IC50 = 1 nM T15497 C39ILN 68259031 IC50 = 50 nM T15497 CKM76G 68259032 IC50 = 40 nM T15497 C0WB3O 68259039 IC50 = 12 nM T15497 C8NBR9 68259112 IC50 = 140 nM T15497 CFHM61 68318287 IC50 = 130 nM T15497 C3Z8UY 68329608 IC50 = 150 nM T15497 CVM9Q1 68503758 IC50 > 25000 nM T15497 CA15ND 68505312 IC50 > 25000 nM T15497 C0US2T 68505327 IC50 > 25000 nM T15497 CX8W7F 68508048 IC50 > 25000 nM T15497 C01YOJ 71452690 Ki = 4900 nM T15497 CQ5E0J 71455094 Ki = 20260 nM T15497 COK0V6 71458757 Ki = 68625 nM T15497 C74PUE 71462285 Ki = 15990 nM T15497 C8XJ0I 71733818 IC50 > 25000 nM T15497 CXC78L 71733909 IC50 > 25000 nM T15497 C7B5XE 71733910 IC50 > 25000 nM T15497 CQ21ZD 71733911 IC50 > 25000 nM T15497 CZG0S2 71733912 IC50 > 25000 nM T15497 CD3Y5K 72543866 IC50 = 500 nM T15497 CQTJ82 72547455 IC50 = 84 nM T15497 C4G2UR 72695027 Ki > 17500 nM T15497 CDFO42 72695136 Ki > 17500 nM T15497 CWTO83 91810751 Ki > 17500 nM T15497 CR4DE7 118175009 Ki > 19500 nM T15497 CSJ4A9 118352160 EC50 > 10000 nM T15497 CE6L8I 118352177 EC50 > 10000 nM T15497 C8PKA7 118352211 EC50 > 10000 nM T15497 CPS7M4 118352285 EC50 > 10000 nM T15497 C7Z3HU 122180289 IC50 > 30000 nM T15497 C2NG1J 122180295 IC50 > 30000 nM T15497 C8ZRJ0 126495398 EC50 = 4200 nM T15497 C8SRZ5 126495427 EC50 > 10000 nM T15497 CD72CT 126495432 EC50 > 10000 nM T15497 CN72WL 126495463 EC50 = 97 nM T15497 CV1A6C 126495491 EC50 = 970 nM T15497 CYP3E5 126495507 EC50 > 10000 nM T15497 C2N7XJ 127026652 Ki = 8418 nM T15497 CX9M6D 127029402 EC50 > 10000 nM T15497 CWXR72 127029417 Ki > 50000 nM T15497 CW1O4F 127029692 EC50 > 10000 nM T15497 CBCQ64 127047601 Ki > 10000 nM T15497 CTR62O 127052613 EC50 = 1.4 nM T15497 CGZR45 127052614 EC50 = 160 nM T15497 COVY75 127052615 EC50 = 700 nM T15497 CZT3E1 135581997 IC50 = 50.12 nM T15497 CY4OI9 136003254 IC50 = 140 nM T15497 CA8QC3 141730897 IC50 > 10000 nM T15497 C2P9GV 141730900 IC50 > 10000 nM T15497 CK6E7L 141730914 IC50 > 10000 nM T15497 C7B5WG 141730916 IC50 > 10000 nM T15497 C62DUY 141730923 IC50 > 10000 nM T15497 C3YR5W 145961578 IC50 = 12 nM T15497 C9VP2I 145963362 IC50 = 12 nM T15497 CGV2E8 145977227 EC50 = 2000 nM T15497 CDN70S 146014480 IC50 > 10000 nM T15497 CZ10RG 155522808 IC50 > 10000 nM T15497 C7UY3Q 155529786 IC50 > 10000 nM T15497 C82RVN 155554217 IC50 > 10000 nM T15497 D02LXJ 9813912 Ki > 100000 nM T15497 D02MXT 24952929 Ki > 5600 nM T15497 D02SAD 44419388 Ki > 100000 nM T15497 D03OYD 5311240 IC50 = 1360 nM T15497 D07JMB 44289922 Ki > 100000 nM T15497 D07UDT 15551229 Ki = 39000 nM T15497 D08MNO 25886893 Ki > 10000 nM T15497 D08ZYC 11595431 Ki < 1584.89 nM T15497 D0H5TU 11524454 IC50 > 20000 nM T15497 D0J9PG 119461 Ki = 1200 nM T15497 D0O9ES 5311053 IC50 = 496 nM T15497 D0R2TW 10238338 IC50 = 2.512 nM T15497 D0S2LO 9864831 Ki > 13000 nM T15497 D0S6NE 11306423 Ki = 4 nM T15497 D0TA0L 23685469 Ki > 1000 nM T15497 D0Y1IF 23664784 Ki > 1000 nM T15497 D0Z3XJ 9817405 Ki > 100000 nM T01777 D01AZG 5073 Ki = 3.2 nM T01777 D01JGV 441975 Ki = 5 nM T01777 D01JUF 5775 Ki = 8.4 nM T01777 D03MIR 3157 Ki = 280 nM T01777 D03SKR 2803 Ki = 9.333 nM T01777 D04JEE 4946 EC50 > 5011.87 nM T01777 D05MBZ 129211 Ki = 7.9 nM T01777 D05ZIK 4205 Ki = 18 nM T01777 D06OFS 68712 Ki = 12.59 nM T01777 D07MOX 439260 Ki = 63 nM T01777 D09EBS 4636 Ki = 1 nM T01777 D0AE3X 2435 EC50 = 3.4 nM T01777 D0CQ0Z 33630 Ki = 445 nM T01777 D0E9PK 4810 Ki = 2000 nM T01777 D0G8NN 119570 Ki = 52.2 nM T01777 D0H3HM 60795 Ki = 100 nM T01777 D0H4JM 8969 Ki = 0.5 nM T01777 D0H7KF 5002 Ki = 100 nM T01777 D0K0MW 30668 EC50 = 1.38 nM T01777 D0MT0M 2216 Ki = 30 nM T01777 D0O6IZ 4436 Ki = 2.291 nM T01777 D0P9RF 5401 Ki = 78 nM T01777 D0R6RO 4184 Ki = 3.8 nM T01777 D0U3DU 5311068 Ki = 30.9 nM T01777 D0V4QS 135398745 Ki = 82 nM T01777 D0WV3U 4893 Ki = 24 nM T01777 D0Z1RV 135398737 Ki = 2.9 nM T01777 D05LGX 213041 Ki = 13.8 nM T01777 D0LI1C 44469321 IC50 > 10000 nM T01777 D0N1HW 5311200 Ki = 230 nM T01777 D00OWF 5280953 Ki = 810 nM T01777 D02LHR 33625 Ki = 476 nM T01777 D02ZSU 9838763 EC50 = 1995.26 nM T01777 D03QMR 5685 Ki = 0.8 nM T01777 D05FYA 3035905 Ki = 346.74 nM T01777 D05OVC 71310 Ki = 4.169 nM T01777 D08OWQ 122295 Ki = 64 nM T01777 D0B1MJ 6918097 Ki = 450 nM T01777 D0BC6Q 9837551 Ki = 8.9 nM T01777 D0K9JP 9928332 Ki = 2.1 nM T01777 D0L5TJ 10527469 Ki = 16.6 nM T01777 D0N7LZ 126225 Ki = 21 nM T01777 D0OU7P 1242 Ki = 83.18 nM T01777 C4JQ7T 2068 Ki > 20000 nM T01777 C5H9CN 9287 Ki > 10000 nM T01777 CL3T5Z 27013 Ki < 100 nM T01777 COY1P0 32238 Ki = 15135.61 nM T01777 CNZD18 36381 Ki = 682 nM T01777 CU86VK 54459 Ki = 17.78 nM T01777 C28VFY 60602 Ki = 330 nM T01777 C2H1VA 131829 EC50 = 104.71 nM T01777 CLK7P3 169713 IC50 > 10000 nM T01777 CF4V5Q 185076 EC50 = 14.13 nM T01777 C09JTU 199798 Ki = 862 nM T01777 CH6WT3 218362 EC50 = 2.188 nM T01777 C9P2AL 286547 Ki = 239.88 nM T01777 CQ5Z8Y 294234 Ki = 33.11 nM T01777 CU0O7M 434526 Ki = 645.65 nM T01777 CFUJ25 737253 Ki = 1513.56 nM T01777 CZN6S9 743974 EC50 > 31622.78 nM T01777 CXJA39 770500 Ki = 15488.17 nM T01777 C8XW6S 1393724 Ki = 11.75 nM T01777 CAQ2J0 3034396 Ki = 2320 nM T01777 CS2Q1G 3045401 IC50 = 1.698 nM T01777 CU4T6Q 3086326 EC50 = 30.9 nM T01777 CJ6D8N 3342390 Ki < 1000 nM T01777 C1WCM4 4306793 Ki = 15488.17 nM T01777 C8HYF7 4657799 Ki = 8317.64 nM T01777 C8ZBJ9 7059292 Ki = 5011.87 nM T01777 CK3NP7 8032110 Ki = 537.03 nM T01777 CHD32K 9794524 Ki = 340 nM T01777 C4K7ZJ 9795515 Ki = 88 nM T01777 C5Z2KM 9805944 Ki = 2.4 nM T01777 C9PZN8 9815633 Ki = 172 nM T01777 C5A8UR 9815707 EC50 = 4.074 nM T01777 CXP87Y 9816063 Ki = 205 nM T01777 C1X0UA 9817256 Ki < 5011.87 nM T01777 CO9VA3 9820671 IC50 > 1000 nM T01777 C6KJ7P 9827677 Ki = 1479 nM T01777 CQZ6I0 9828476 Ki = 81.28 nM T01777 CBN06W 9839050 Ki = 69 nM T01777 CB7L9H 9846548 Ki = 6.2 nM T01777 CY2D5T 9851486 Ki = 371.54 nM T01777 CM13ZV 9856041 IC50 > 30000 nM T01777 CQ2L0J 9859437 EC50 = 110 nM T01777 CV2HW7 9883506 Ki = 12.8 nM T01777 C3DB5H 9884781 Ki = 336 nM T01777 C8HS4Q 9895326 Ki = 190.55 nM T01777 CFI97S 9904205 IC50 = 1862.09 nM T01777 CYWQ50 9906447 Ki > 10000 nM T01777 C7JFZ5 9906978 Ki = 16.4 nM T01777 C7SMT0 9908904 IC50 > 1000 nM T01777 C32ZXG 9923679 Ki = 690 nM T01777 CUQ8I5 9947861 EC50 = 794.33 nM T01777 CO2X8D 9951544 IC50 = 14.13 nM T01777 CF1C5Q 9960497 Ki = 300 nM T01777 C3O9SC 9971924 EC50 = 60.26 nM T01777 CC05RX 9982218 Ki = 100 nM T01777 CQL12P 10004545 Ki > 2000 nM T01777 C52JBP 10028898 Ki = 0.8 nM T01777 C2EUY0 10035109 Ki > 10000 nM T01777 C3Z4OD 10040286 Ki > 10000 nM T01777 C5MZ6I 10042547 Ki > 10000 nM T01777 C7D0GO 10044968 Ki = 15 nM T01777 CB82XU 10045088 Ki = 7.499 nM T01777 C3MTF4 10045713 Ki = 2.3 nM T01777 C4PCO3 10065083 Ki = 80 nM T01777 CZ0U2N 10070896 Ki = 5 nM T01777 COF5U3 10109188 Ki = 25 nM T01777 C9XCB3 10132386 Ki = 34.99 nM T01777 CE27RV 10135864 EC50 > 10000 nM T01777 CRS5B6 10176999 EC50 = 6.6 nM T01777 CNB56M 10177445 Ki = 52 nM T01777 CQ8HX2 10198135 Ki = 512 nM T01777 C7MKP9 10199335 EC50 = 1995.26 nM T01777 CC2KV3 10214826 Ki > 10000 nM T01777 CLY2B9 10220232 Ki = 26 nM T01777 CU2B9P 10221004 Ki = 2511.89 nM T01777 CX9YD5 10221005 EC50 = 1122.02 nM T01777 CVF1E5 10246054 IC50 > 1000 nM T01777 C0LOA6 10251036 Ki = 5.9 nM T01777 C6G0AY 10266032 EC50 = 26.92 nM T01777 CBE9K1 10317643 Ki = 42.95 nM T01777 C4MD0S 10318507 Ki = 8.299 nM T01777 CSU1R6 10319299 Ki = 34.99 nM T01777 C6W5DM 10333157 EC50 = 18.62 nM T01777 CLG82T 10356463 Ki > 10000 nM T01777 COS13I 10362866 Ki = 5 nM T01777 C4H6YF 10379435 EC50 = 3162.28 nM T01777 CDAC63 10381889 IC50 = 870.96 nM T01777 C3N7TF 10382537 EC50 = 54.95 nM T01777 CIQ02H 10436842 Ki = 3846 nM T01777 CIDE58 10473701 Ki = 5.395 nM T01777 C8FA2T 10474679 Ki = 6.397 nM T01777 CBS8U6 10475736 Ki = 50 nM T01777 CW81LP 10480357 Ki = 0.3 nM T01777 CJ0K1T 10507651 Ki = 407.38 nM T01777 C2U8AC 10508016 Ki = 630.96 nM T01777 C4XZ3Y 10508132 Ki = 812.83 nM T01777 CZP09X 10508332 Ki = 398.11 nM T01777 C4X9EF 10531532 Ki = 245.47 nM T01777 C7MI2N 10531766 Ki = 575.44 nM T01777 CF24MW 10579368 Ki = 776.25 nM T01777 CK8SO7 10603951 Ki = 245.47 nM T01777 C1DXO0 10609673 Ki = 1500 nM T01777 CB26QH 10626982 Ki = 478.63 nM T01777 CSWC40 10627021 Ki = 416.87 nM T01777 CF1P6Z 10651080 Ki = 724.44 nM T01777 C3K7UP 10651654 Ki = 158.49 nM T01777 CTB7L2 10674896 Ki = 870.96 nM T01777 CTSY18 10682720 Ki = 290 nM T01777 C3IX8A 10707358 Ki = 10.72 nM T01777 CT1K3B 10769331 Ki = 47.86 nM T01777 C3O7YN 10793665 Ki = 1000 nM T01777 C0D6MW 10793963 Ki = 281.84 nM T01777 CBO8N9 10818003 Ki = 426.58 nM T01777 CE80NV 10841190 Ki = 1148.15 nM T01777 CYSL64 10841387 Ki = 323 nM T01777 C5AY9R 10848826 Ki = 66.07 nM T01777 C8VT6G 10916464 Ki = 3981.07 nM T01777 CH95TI 10923927 Ki = 2691.53 nM T01777 C3CI6Z 10934575 EC50 = 8.913 nM T01777 CGW87Y 11034737 EC50 = 7.943 nM T01777 CA7IB5 11043720 EC50 = 112.2 nM T01777 C48QYR 11058166 EC50 = 446.68 nM T01777 C7JI1M 11059195 Ki < 5011.87 nM T01777 C7R2AZ 11079593 Ki < 5011.87 nM T01777 C91BKL 11090351 Ki = 257.04 nM T01777 CFE1M7 11097789 EC50 = 100 nM T01777 CTG4I5 11098175 Ki = 602.56 nM T01777 CR6K4V 11109088 EC50 = 2.818 nM T01777 C6SXJ0 11140033 EC50 = 93.33 nM T01777 CG40BP 11140345 EC50 = 15.85 nM T01777 CO0XW1 11140347 EC50 = 5.623 nM T01777 CTA5J4 11173544 Ki = 251.19 nM T01777 CU86DN 11173568 Ki = 309.03 nM T01777 C5JYO7 11186227 Ki = 331.13 nM T01777 C0W4SM 11186523 Ki = 93 nM T01777 C1VIN4 11190988 Ki = 0.5 nM T01777 CHU5B0 11191321 Ki = 1.6 nM T01777 C3ALW8 11199581 Ki = 1621.81 nM T01777 C9T7YZ 11199593 Ki = 707.95 nM T01777 C01AFD 11200476 Ki = 4.5 nM T01777 C5YQ0F 11203101 Ki = 0.65 nM T01777 C62KQF 11211035 Ki = 16.98 nM T01777 CYQ65M 11214030 Ki = 0.2 nM T01777 CEGZ35 11221758 Ki = 1230.27 nM T01777 CV2R8E 11224953 Ki = 2.7 nM T01777 C59VOU 11225732 Ki = 18 nM T01777 C3RO9W 11225779 Ki = 0.2 nM T01777 COCU26 11246610 Ki = 302 nM T01777 CXNM72 11259744 Ki = 0.2 nM T01777 C5PWC6 11260018 Ki = 0.5 nM T01777 CNTE30 11265631 EC50 = 39.81 nM T01777 CZ8DY9 11271808 Ki = 0.1 nM T01777 C8SYW5 11277479 Ki = 245.47 nM T01777 C84NSM 11278634 Ki < 10000 nM T01777 CNAQ56 11293787 Ki = 11 nM T01777 CA1D3O 11300487 Ki = 234.42 nM T01777 C7VS0M 11306100 Ki = 0.03 nM T01777 CM67PT 11318438 Ki = 0.5 nM T01777 CG8JA6 11333552 Ki = 10471.29 nM T01777 C3JBI0 11338418 Ki > 500 nM T01777 C96OKG 11346584 Ki = 17.78 nM T01777 CV17WA 11360447 EC50 = 58.88 nM T01777 CI69GW 11361608 EC50 = 100 nM T01777 CA28SQ 11371902 EC50 = 93.33 nM T01777 C9U5WT 11380132 Ki = 1258.93 nM T01777 C1ZOY6 11380133 Ki = 1445.44 nM T01777 C4JVS8 11385652 Ki = 9.8 nM T01777 CB01AS 11448533 Ki = 5888.44 nM T01777 CX8CN6 11473729 Ki = 5888.44 nM T01777 CP5RO3 11564613 Ki = 562.34 nM T01777 CZA0M9 11653915 Ki = 3.8 nM T01777 CJ1KW9 11741010 Ki = 132 nM T01777 CPG15O 11743399 IC50 > 1000 nM T01777 CIM1E0 11750482 Ki = 8 nM T01777 CX7TO1 11785068 Ki = 0.3 nM T01777 CE4Q9W 11785961 Ki = 0.2 nM T01777 CFTI34 11801828 Ki = 1023.29 nM T01777 C1VWL5 11811395 Ki < 5011.87 nM T01777 CXLW54 11948707 Ki = 109 nM T01777 C8JQL7 11957735 IC50 > 10000 nM T01777 CWA2B6 12304323 Ki = 4063 nM T01777 CIUR20 12699315 Ki = 5754.4 nM T01777 C2V9FL 13091268 Ki = 142.8 nM T01777 CWBX46 13123534 EC50 = 223.87 nM T01777 CP90IU 13178306 Ki = 72.44 nM T01777 C1CX2S 15675860 Ki = 645.65 nM T01777 CXM74T 16090594 Ki = 83.95 nM T01777 C8QLC1 16090595 Ki = 8.299 nM T01777 C01RFM 16090596 Ki = 6.9 nM T01777 CAYX52 16090597 Ki = 389.94 nM T01777 CW0U8R 16090598 Ki = 134.9 nM T01777 C06KXJ 16090599 Ki = 770 nM T01777 COB96N 16090600 Ki = 100 nM T01777 C6YPM3 16090601 Ki = 8.995 nM T01777 CR02MW 16090602 Ki = 9.2 nM T01777 CC5HV2 16090621 Ki = 34.99 nM T01777 COTF82 16090622 Ki = 8.492 nM T01777 CB2Z6H 16090623 Ki = 7.691 nM T01777 C4WAZ1 16090624 Ki = 76 nM T01777 C6MH3Z 16090625 Ki = 87 nM T01777 CX98OC 16090626 Ki = 16 nM T01777 C6D0WK 16090627 Ki = 82 nM T01777 C1B5TL 16090628 Ki = 8.492 nM T01777 CTXU32 16090630 Ki = 3.8 nM T01777 CD8FX2 16090631 Ki = 4.898 nM T01777 C63QEJ 16090632 Ki = 205 nM T01777 C98XNF 16090633 Ki = 38 nM T01777 C1G7KL 16090634 Ki = 769.13 nM T01777 C8YBI4 16090635 Ki = 109.9 nM T01777 CERP08 16219807 Ki < 10000 nM T01777 CNF70V 16220269 IC50 = 10400 nM T01777 CZ2IS9 16660294 Ki > 10000 nM T01777 CVU96E 16725934 Ki = 20 nM T01777 CFMX86 16757089 EC50 = 10 nM T01777 C6OJ3A 16757182 Ki = 537.03 nM T01777 C6AOE8 19426635 IC50 > 1000 nM T01777 CPRJ25 21392988 Ki = 16595.87 nM T01777 C3T5HF 21509921 Ki = 173 nM T01777 CT7XG9 21830793 Ki = 15 nM T01777 C8GUJ3 22120322 IC50 = 1.288 nM T01777 CGO3B8 22120332 IC50 = 0.7079 nM T01777 C02AEX 22493245 Ki = 2630.27 nM T01777 CF9D1U 23622576 EC50 = 20.89 nM T01777 CDC91N 24839550 Ki = 891.25 nM T01777 CY21RE 24841480 Ki = 830 nM T01777 C2C7WN 24882007 Ki = 640 nM T01777 C8WH5Z 24906160 EC50 = 501.19 nM T01777 C3RQ1P 24906196 Ki = 338.84 nM T01777 CBT65R 24906197 Ki = 676.08 nM T01777 C9OAG1 24906198 EC50 = 50.12 nM T01777 CYL83G 24906199 EC50 = 10 nM T01777 CC9W0R 24906200 Ki = 204.17 nM T01777 CYEA86 24906201 EC50 = 794.33 nM T01777 CIR8G1 24906202 Ki = 1584.89 nM T01777 CPH75D 24906203 Ki = 1258.93 nM T01777 CBUH25 24906241 Ki = 691.83 nM T01777 C7Y2SB 24906243 Ki = 245.47 nM T01777 C1VRJ3 25014630 IC50 = 11000 nM T01777 C2G1JK 25053351 Ki = 77.6 nM T01777 C9XMH7 25110718 Ki = 0.9 nM T01777 CX04LB 25142456 Ki = 2 nM T01777 C4MRQ0 27842480 Ki = 2841 nM T01777 CWT9F7 28918670 EC50 = 97.72 nM T01777 CAM63X 42618195 IC50 > 1000 nM T01777 C8K4UF 42618197 IC50 > 1000 nM T01777 CJ3NP5 42636941 IC50 = 741.31 nM T01777 CMV4E2 42656257 Ki = 13803.84 nM T01777 CE7C3O 42669828 Ki = 22387.21 nM T01777 CVG6X1 44209472 Ki = 194.5 nM T01777 CD5AB7 44209480 Ki = 308.2 nM T01777 C9O1RI 44215744 Ki = 3.1 nM T01777 CO65VL 44269006 EC50 = 61.66 nM T01777 C0TP2Z 44269013 EC50 = 154.88 nM T01777 CW6A9E 44269089 EC50 = 398.11 nM T01777 CZ63DE 44269122 Ki = 263.03 nM T01777 CDS8G5 44269140 EC50 = 100 nM T01777 CE20CZ 44275807 Ki = 1621.81 nM T01777 CZ5P6U 44288769 Ki = 1905 nM T01777 CZ7O4D 44288847 Ki = 4677 nM T01777 C6DYQ1 44288874 Ki = 1995 nM T01777 CAG7E1 44288877 Ki = 6531 nM T01777 CQ3Y5R 44288945 Ki = 313 nM T01777 C5ZL4A 44289035 Ki = 1096 nM T01777 CLRZ30 44292232 EC50 = 21.38 nM T01777 C7GUL1 44292381 Ki = 52.48 nM T01777 C3G1KO 44292385 EC50 = 13.8 nM T01777 C0R8WU 44292386 EC50 = 1.995 nM T01777 C6G8ZC 44311789 Ki = 11481.54 nM T01777 C5L1WN 44312036 Ki = 645.65 nM T01777 CT46CK 44312037 Ki = 28183.83 nM T01777 C3XFH4 44312198 Ki = 48977.88 nM T01777 CZ4TN0 44314198 EC50 = 4.074 nM T01777 CCI07K 44314200 EC50 = 24.55 nM T01777 CV8WZ0 44318454 IC50 = 1174.9 nM T01777 CXJL56 44318842 IC50 > 1000 nM T01777 CA56FM 44324725 Ki = 1.9 nM T01777 CW16JD 44324737 Ki = 0.8 nM T01777 CA84SN 44324765 Ki = 0.5 nM T01777 COA3H4 44324800 Ki = 0.1 nM T01777 CK32IL 44324859 Ki = 4.7 nM T01777 CMB1S6 44324860 Ki = 89 nM T01777 C8HUD2 44324887 Ki = 2.3 nM T01777 CCT53K 44324900 Ki = 89 nM T01777 CL1F3T 44324906 Ki = 1.9 nM T01777 CPAL75 44324937 Ki = 1.7 nM T01777 CY04JW 44324972 Ki = 0.2 nM T01777 C76UJT 44325027 Ki = 30 nM T01777 C1RS8C 44325028 Ki = 89 nM T01777 CR4Q1C 44325038 Ki = 36 nM T01777 C4SZJ2 44325044 Ki = 13 nM T01777 CQX1Y0 44325049 Ki = 0.6 nM T01777 C0N3JG 44325050 Ki = 0.2 nM T01777 CEYD96 44325075 Ki = 5.3 nM T01777 CGS4E7 44325079 Ki = 89 nM T01777 CV7L8H 44330114 Ki = 0.4 nM T01777 C7Q1HP 44330168 Ki = 0.2 nM T01777 COY19U 44330368 Ki = 0.6 nM T01777 C1Z6DB 44330369 Ki = 0.3 nM T01777 CKO67I 44330427 Ki = 0.7 nM T01777 CP7Y9I 44330571 Ki = 9.5 nM T01777 C3AY4O 44330584 Ki = 2.8 nM T01777 CVTA63 44330598 Ki = 0.7 nM T01777 C83NZA 44330609 Ki = 23 nM T01777 C2AOH6 44330617 Ki = 0.2 nM T01777 C2RQ3Z 44330621 Ki = 10 nM T01777 C7JP2X 44330635 Ki = 0.4 nM T01777 CCVE83 44330645 Ki = 0.5 nM T01777 CO8XC7 44330653 Ki = 0.2 nM T01777 C47ZPQ 44330668 Ki = 0.2 nM T01777 CGJ05Y 44330679 Ki = 2.1 nM T01777 C9D2SN 44330857 Ki = 0.9 nM T01777 CZ2X3A 44352155 EC50 = 147.91 nM T01777 C67ZNM 44352207 EC50 = 57.54 nM T01777 C6KJV8 44371744 EC50 = 56.23 nM T01777 CI90WF 44371745 EC50 = 100 nM T01777 C09ADW 44371755 EC50 = 27.54 nM T01777 C76VTG 44371864 EC50 = 27.54 nM T01777 C3K6GE 44376845 IC50 = 57.54 nM T01777 CPD18R 44376900 IC50 = 1.622 nM T01777 CE46SW 44376923 IC50 = 1.072 nM T01777 C7UW8Z 44376927 IC50 = 3.631 nM T01777 C8GT5O 44376936 IC50 = 6.607 nM T01777 CLC2T4 44376954 IC50 = 0.8511 nM T01777 C9IPC3 44376958 IC50 = 1.202 nM T01777 CX4A1Z 44376975 IC50 = 2.692 nM T01777 C14SMK 44376984 IC50 = 0.6166 nM T01777 C0V4XL 44376993 IC50 = 1.349 nM T01777 CX0UR3 44377006 IC50 = 27.54 nM T01777 CB2R0M 44377007 IC50 = 2.239 nM T01777 C2ID6U 44377035 IC50 = 1.318 nM T01777 C6R9OZ 44377036 IC50 = 0.7244 nM T01777 C97QIG 44377200 IC50 = 0.6918 nM T01777 C93JCM 44387789 Ki = 0.2 nM T01777 CI52GK 44387798 Ki = 11 nM T01777 CX7O9S 44401041 Ki = 200 nM T01777 C5XC2B 44401042 Ki = 677 nM T01777 CD56EA 44401105 Ki = 742 nM T01777 CW3PC2 44401106 Ki = 78 nM T01777 C9WH7P 44401164 Ki = 59 nM T01777 C9CWX1 44401194 Ki = 219 nM T01777 CXT84G 44401243 Ki = 26 nM T01777 CFM28R 44402344 Ki = 19 nM T01777 CX6NT4 44402345 Ki = 2.8 nM T01777 CN5P3Z 44402346 Ki = 1.1 nM T01777 C6W9BU 44402352 Ki = 32 nM T01777 CUA7D5 44402477 Ki = 8.5 nM T01777 CD8A6C 44402531 Ki = 5.2 nM T01777 C9S8WN 44402579 Ki = 8 nM T01777 CW4NO7 44402583 Ki = 3 nM T01777 CI47TG 44421258 EC50 = 2691.53 nM T01777 CK7HF3 44424855 Ki = 4.5 nM T01777 C28OZL 44438147 Ki = 19 nM T01777 CKB9O7 44438148 Ki = 9.6 nM T01777 C1AR8P 44438152 Ki = 19 nM T01777 CZR64Y 44438161 Ki = 9.4 nM T01777 CG38YN 44438165 Ki = 9.4 nM T01777 C8RC7O 44438166 Ki = 4.2 nM T01777 C5GPZ7 44438167 Ki = 0.8 nM T01777 C0QI8L 44438168 Ki = 3.5 nM T01777 CZL97F 44455426 Ki = 148 nM T01777 C12XGE 44456400 Ki = 794.33 nM T01777 CQ2IX7 44461606 IC50 > 1000 nM T01777 C4LUK7 44549156 EC50 = 39.81 nM T01777 CVA67X 44568347 Ki = 600 nM T01777 C8N3ID 44568614 Ki = 64.57 nM T01777 CWM4U7 44579184 Ki = 23 nM T01777 CLO8A9 44579185 Ki = 5 nM T01777 CGVM03 44579186 Ki = 3 nM T01777 CM6L2Y 44579187 Ki = 0.8 nM T01777 CBDL39 44579228 Ki = 0.5 nM T01777 CX5O1H 44579229 Ki = 0.8 nM T01777 C3G5YK 44579230 Ki = 0.6 nM T01777 CKTJ23 44579231 Ki = 15.7 nM T01777 C57BWM 44579271 Ki = 2.5 nM T01777 C7R9XM 44579272 Ki = 1.7 nM T01777 CZY26H 44579303 Ki = 9.2 nM T01777 CEJ4R8 44582676 Ki = 333 nM T01777 C5QB4K 44582678 Ki = 143 nM T01777 C01RCI 44582705 Ki = 154 nM T01777 CWO70X 45260703 Ki < 5011.87 nM T01777 C4VOW6 45260704 EC50 = 28.18 nM T01777 CQ0R5Y 45264581 EC50 = 5.623 nM T01777 C39CDN 45264638 EC50 = 28.18 nM T01777 C0CHF4 45482789 IC50 = 215 nM T01777 CQHW85 45487089 EC50 = 63.1 nM T01777 CI34PT 45487144 Ki = 263.03 nM T01777 CC9GH0 45487145 EC50 = 50.12 nM T01777 C7MZ9Y 45487955 EC50 = 25.12 nM T01777 CLW5M9 45487956 EC50 = 39.81 nM T01777 C45DAV 45487958 Ki = 501.19 nM T01777 CZSW97 45487962 EC50 = 154.88 nM T01777 C34ZXM 46225029 Ki = 20 nM T01777 C1WT4J 46743607 Ki = 5248.07 nM T01777 C1C6WH 46743614 Ki = 7244.36 nM T01777 C03LTM 46869265 Ki = 1100 nM T01777 CJ6K2R 46891598 Ki = 4.5 nM T01777 C8VUO2 49781004 Ki = 66.07 nM T01777 C0LAT9 49781005 Ki = 1.95 nM T01777 C12UVE 49781006 Ki = 10.23 nM T01777 CW1V4K 49781007 Ki = 1.549 nM T01777 CF9L7Z 49781008 Ki = 89.13 nM T01777 CQ2EN5 49781222 Ki = 0.537 nM T01777 CV62OU 49781223 Ki = 1.259 nM T01777 C3I5HP 49781224 Ki = 1.479 nM T01777 CF5CO4 49781228 Ki = 0.1288 nM T01777 CW5X6A 49781887 Ki = 2.138 nM T01777 C2LZJ0 49783209 Ki = 556 nM T01777 C57SMG 49783415 Ki = 989 nM T01777 C0TG6I 49783419 Ki = 593 nM T01777 C28CKM 49836301 EC50 = 25.12 nM T01777 C5JO6E 49836302 Ki = 177.83 nM T01777 C9TNO4 49836303 EC50 = 35.48 nM T01777 CL6QA1 49836304 Ki = 125.89 nM T01777 CE1S9B 49836305 EC50 = 6.31 nM T01777 CP0DJ4 49836306 EC50 = 100 nM T01777 CJM3F9 49836307 Ki = 112.2 nM T01777 C0LN3I 49836308 EC50 = 25.12 nM T01777 C2RY0J 50878551 Ki = 501.19 nM T01777 C1W6TV 50898777 Ki > 10000 nM T01777 CXMZ73 50898778 Ki > 10000 nM T01777 CE4KP1 51050257 Ki > 10000 nM T01777 CR8MI3 52941512 Ki = 0.2951 nM T01777 CZ4SA1 52942940 Ki = 4265.8 nM T01777 CH3YE5 52943739 Ki = 2.818 nM T01777 C70LBS 52944548 Ki = 0.1698 nM T01777 C7WN4S 52948958 Ki = 0.4365 nM T01777 C5W7SH 52950140 Ki = 1.175 nM T01777 CB37XF 53325861 Ki = 2071 nM T01777 CJKO58 56852956 Ki = 125.89 nM T01777 CB0P9N 56944383 Ki = 1.9 nM T01777 C1TC7Q 56963799 Ki > 10000 nM T01777 C4RBY6 57345625 EC50 = 165.96 nM T01777 C1US6F 57345626 EC50 = 10 nM T01777 CNU83J 57345627 EC50 = 114.82 nM T01777 CD50GK 57345628 EC50 = 1.995 nM T01777 C4FA1T 57345629 EC50 = 47.86 nM T01777 CO2W7Z 57384051 Ki > 10000 nM T01777 C80DHR 57393066 Ki > 10000 nM T01777 C4N0TW 57393922 EC50 = 630.96 nM T01777 C6X0ZI 57394788 Ki > 10000 nM T01777 CR6U3P 57394789 Ki > 10000 nM T01777 CH84EC 57395663 EC50 = 794.33 nM T01777 CL37YV 57395731 EC50 = 199.53 nM T01777 C5I3DG 57395732 EC50 = 79.43 nM T01777 CR1Y7M 57398332 Ki > 10000 nM T01777 CM9WK5 57399145 Ki = 758.58 nM T01777 CIB2L3 57399991 Ki > 10000 nM T01777 CQ7MC1 57400959 EC50 = 316.23 nM T01777 CZX05B 57401706 Ki = 45.1 nM T01777 C9WE2A 57401787 Ki = 6165.95 nM T01777 C56WAY 57402717 Ki = 831.76 nM T01777 C1BFP4 57402718 EC50 = 100 nM T01777 CP21KC 57403508 Ki = 7413.1 nM T01777 C3XL7O 66561967 Ki = 4264 nM T01777 CLM79R 70686398 Ki > 10000 nM T01777 CJQX48 70693375 Ki = 234.42 nM T01777 CST13M 70695474 EC50 = 1.995 nM T01777 C6CNI0 70696790 Ki > 10000 nM T01777 CKD60A 70789640 Ki = 575 nM T01777 CC43QK 71151588 Ki = 190 nM T01777 C6DU5P 71450548 Ki = 1369 nM T01777 C9VZ8J 71450550 Ki = 533 nM T01777 CGQ0R2 71450907 Ki = 1.7 nM T01777 CTDN12 71452341 Ki = 249 nM T01777 C4NDR3 71452382 Ki = 1704 nM T01777 C6ZWV2 71452383 Ki = 1874 nM T01777 CYK20Z 71452384 Ki = 1835 nM T01777 CDTW09 71452387 Ki = 1783 nM T01777 C6G2HC 71455894 Ki = 1145 nM T01777 CUX98O 71456238 Ki = 4 nM T01777 COG3Y0 71456239 Ki = 112 nM T01777 CYR3D4 71456240 Ki = 3.9 nM T01777 CP7JI0 71457691 Ki = 699 nM T01777 CK5T4P 71459604 Ki = 557 nM T01777 C1CD2B 71461344 Ki = 4732 nM T01777 CR3LH2 71461647 Ki = 6.3 nM T01777 CL91AC 71463022 Ki = 1542 nM T01777 CKX5O8 71463061 Ki = 4347 nM T01777 C1Y9IC 71463063 Ki = 1491 nM T01777 C5L8NJ 72947314 EC50 = 234.42 nM T01777 CE1JY2 72947315 Ki = 794.33 nM T01777 CC65OA 73213195 Ki = 770 nM T01777 CW83DK 73213196 Ki = 446 nM T01777 C02FTM 73291731 EC50 = 25.12 nM T01777 CCV91B 73346042 Ki = 173.7 nM T01777 CRG9J8 73346332 Ki = 5048 nM T01777 C6J0TM 73346336 Ki = 2793 nM T01777 CC35AI 73347827 Ki = 4738 nM T01777 CW8A0Y 73349359 Ki = 2283 nM T01777 C6BS5L 73349361 Ki = 865 nM T01777 CY2IB5 73349362 Ki = 3727 nM T01777 CV1U7L 73352414 Ki = 1510 nM T01777 C87LGB 73352415 Ki = 3980 nM T01777 C1NJ0R 73353884 Ki = 3081 nM T01777 C4F7VK 73355415 Ki = 683 nM T01777 C81CIL 73355418 Ki = 993 nM T01777 C10ASZ 73355420 Ki = 2520 nM T01777 C8IDL3 75306277 Ki = 31.62 nM T01777 CUQ6V0 92042918 Ki < 1000 nM T01777 C7YQM3 101333429 Ki = 560 nM T01777 CCY5S0 118717248 Ki = 600 nM T01777 CCR09Q 118717249 Ki = 1200 nM T01777 CTE58Z 118730369 Ki = 200 nM T01777 C4G3YC 118734875 Ki = 1500 nM T01777 C9AIE1 118734876 Ki = 1800 nM T01777 CK4ER0 122180567 Ki = 1071.52 nM T01777 C5X8MN 122186880 Ki = 433 nM T01777 C7ODW3 122195524 Ki > 900 nM T01777 CTBN56 127026052 Ki = 794.33 nM T01777 C8MC1I 127028408 Ki = 275.42 nM T01777 CR61YN 127034912 Ki < 100 nM T01777 CZ61LK 127034966 EC50 > 5011.87 nM T01777 CA0SN5 127034967 EC50 > 5011.87 nM T01777 CQ0ZT9 127035062 Ki = 429 nM T01777 CU49VE 127036186 Ki = 1096.48 nM T01777 CG06BD 127036932 Ki = 630.96 nM T01777 CVW71O 127036953 Ki = 398.11 nM T01777 C4RV9T 129928082 EC50 = 21.88 nM T01777 C1RI8Q 132060720 Ki = 2879 nM T01777 C0DIF5 132060733 Ki = 2466 nM T01777 CY8B9L 132060743 Ki = 254 nM T01777 C4VNA6 132060746 Ki = 1640 nM T01777 CAVB41 132584404 Ki = 1036 nM T01777 CS3FI6 134137108 EC50 = 114.82 nM T01777 CBU81N 134149168 Ki > 10000 nM T01777 CFG4Y1 134156190 EC50 = 158.49 nM T01777 C2PT4I 135356876 Ki = 1320 nM T01777 CKO6D5 135405894 Ki = 1.6 nM T01777 C7HYA8 135440165 Ki = 0.1 nM T01777 CMK06P 135477797 Ki = 3.6 nM T01777 C1IKQ6 135499867 Ki = 15 nM T01777 CTP2R6 135519400 Ki = 0.1 nM T01777 CA39PK 135519421 Ki = 23 nM T01777 CCBM21 135545454 Ki = 5.4 nM T01777 C5J9BC 136019934 Ki = 0.1 nM T01777 CXA5Y9 136044137 Ki = 12 nM T01777 C0TAI6 136274356 Ki > 1000 nM T01777 CF7S1X 136274357 Ki = 9.6 nM T01777 CE8N4S 137641762 Ki > 10000 nM T01777 CKS5V0 137643541 Ki > 10000 nM T01777 CPCY48 137645406 Ki = 1557 nM T01777 CPI68E 137646281 Ki = 433 nM T01777 CLT73G 137647199 Ki = 619 nM T01777 CR9F3Q 137653203 Ki > 10000 nM T01777 CN2LX1 144852560 Ki = 1490 nM T01777 C6P3SR 153287553 Ki = 1000 nM T01777 CV9G7Z 153287572 Ki > 10000 nM T01777 CO85KL 153287574 Ki > 10000 nM T01777 CUSA24 155519891 Ki > 10000 nM T01777 CB79ZW 155536080 Ki > 10000 nM T01777 CH0VC3 155561439 Ki = 3520 nM T01777 CP9TR0 10324985 Ki = 23.7 nM T01777 C13REG 44471685 Ki > 10000 nM T01777 D00GEE 92766 Ki = 161 nM T01777 D01KAX 135453290 Ki = 4700 nM T01777 D01WWC 16573 Ki > 950 nM T01777 D03DMN 1268096 Ki = 28 nM T01777 D03LDH 10758200 Ki = 19.6 nM T01777 D05GDP 599482 Ki = 1740 nM T01777 D06HHJ 10490084 Ki = 2400 nM T01777 D06QKW 2765 EC50 = 398.11 nM T01777 D06UBB 123981 Ki = 20 nM T01777 D07ICV 3072540 Ki = 36.98 nM T01777 D07JMO 10220337 Ki = 1174.9 nM T01777 D07QCC 10946567 Ki = 35 nM T01777 D08DOG 25130235 Ki = 290 nM T01777 D08KLH 108094 Ki = 0.7943 nM T01777 D09ALJ 5280805 Ki = 9637 nM T01777 D09HJL 10331436 IC50 = 14000 nM T01777 D09RPR 16737207 Ki > 10000 nM T01777 D0A6GK 10489502 Ki = 1100 nM T01777 D0BI4T 53315878 Ki > 10000 nM T01777 D0D8GV 9830741 Ki > 45 nM T01777 D0E3OL 4567175 Ki = 1698.24 nM T01777 D0EO4F 9891167 Ki = 82 nM T01777 D0F0IA 11301655 Ki = 1912 nM T01777 D0FU5E 10220053 Ki = 19 nM T01777 D0H3CW 9839317 Ki = 28 nM T01777 D0I3XA 6422124 Ki = 63.1 nM T01777 D0L5MW 181743 Ki = 181 nM T01777 D0L6JS 9816048 Ki = 120 nM T01777 D0L7IZ 540335 Ki = 27.99 nM T01777 D0LI3J 3080926 Ki = 26915.35 nM T01777 D0M9IC 441082 Ki = 10.47 nM T01777 D0N7UE 10198248 Ki = 1412.54 nM T01777 D0PN9R 16655023 Ki = 0.27 nM T01777 D0Q7ZR 9890547 Ki = 74.7 nM T01777 D0S4VR 10655607 Ki = 400 nM T01777 D0V6DJ 5640 Ki = 131 nM T01777 D0Y0SA 135399666 EC50 = 5660 nM T01777 D0Z7EA 643606 Ki = 1 nM T01777 D0ZC4S 10632290 Ki = 8800 nM T46642 D09JUG 60490 IC50 = 580 nM T46642 D0U5QK 1983 IC50 = 44000 nM T46642 D02AIN 122678117 IC50 = 6.3 nM T46642 D05MCS 44473151 IC50 = 2.9 nM T46642 D05WPQ 6438354 IC50 = 110 nM T46642 D0K2ER 3651377 IC50 = 2.5 nM T46642 D0M0QX 23672584 IC50 = 1.9 nM T46642 CK6VT0 60923 IC50 = 1.6 nM T46642 C8ZC2A 1939738 IC50 = 8800 nM T46642 CB0W6Y 2113616 IC50 > 10000 nM T46642 C07KIA 3248047 IC50 = 4800 nM T46642 CQB41T 3269315 IC50 = 440 nM T46642 CLX42I 3427822 IC50 = 3400 nM T46642 CL9YA6 3499355 IC50 = 700 nM T46642 CGPS21 3558510 IC50 = 2900 nM T46642 CD9T2A 3610995 IC50 = 310 nM T46642 C7NOG8 3718582 IC50 > 10000 nM T46642 C4JX9P 3801708 IC50 = 980 nM T46642 CYS82Q 3809108 IC50 = 3800 nM T46642 CZCS61 3825415 IC50 > 10000 nM T46642 C51ZLQ 4400031 IC50 = 500 nM T46642 CS4F5D 4477730 IC50 = 7200 nM T46642 CZ9E1B 4560409 IC50 = 200 nM T46642 CGMD31 4627406 IC50 = 500 nM T46642 C97TEZ 5225487 IC50 = 4400 nM T46642 C3NO4W 9828630 IC50 = 3 nM T46642 C7EH2G 9873179 IC50 = 10 nM T46642 CLC84P 9873906 IC50 = 7 nM T46642 CZ3SA4 9891815 IC50 = 122 nM T46642 CV4GX8 9915340 IC50 = 5 nM T46642 C1CG2S 9916464 IC50 = 2 nM T46642 C6JF5S 9939089 IC50 = 2 nM T46642 C4R1GL 10507589 IC50 = 760 nM T46642 C8CU4E 10722510 IC50 = 370 nM T46642 C10ETF 10746661 IC50 = 2900 nM T46642 CA8J5Q 10770349 IC50 = 32 nM T46642 CZNK34 10794157 IC50 = 72 nM T46642 C4YME1 11214950 IC50 = 2.8 nM T46642 C2XQI7 11526708 IC50 > 1000 nM T46642 COB0M4 14980539 IC50 = 110 nM T46642 C98AEV 14980542 IC50 = 40 nM T46642 C6OFC1 14980546 IC50 = 19 nM T46642 C3OR9Q 14980547 IC50 = 390 nM T46642 C53AEY 15229443 IC50 = 9.3 nM T46642 CFO6V2 15229452 IC50 = 7 nM T46642 C2ATE4 16223458 IC50 = 0.6 nM T46642 CZ5KW2 16223462 IC50 = 1790 nM T46642 CWJZ50 16223655 IC50 = 4.8 nM T46642 CDG38L 16223656 IC50 = 6.9 nM T46642 C8Y7FL 16223657 IC50 = 1.8 nM T46642 C3O7HD 16223851 IC50 = 9 nM T46642 C7HN3Y 16223853 IC50 = 28 nM T46642 C0D9KR 16223854 IC50 = 4 nM T46642 C65MXS 16224046 IC50 = 299 nM T46642 CFK8M4 16224051 IC50 = 229 nM T46642 C7O3VD 16224255 IC50 = 444 nM T46642 C5L1QM 16224456 IC50 = 0.5 nM T46642 CJ0YK4 16224457 IC50 = 4.8 nM T46642 C0LHO6 16224458 IC50 = 6.6 nM T46642 CX5GT3 16224844 IC50 = 2.1 nM T46642 C29KRC 16225463 IC50 = 3.3 nM T46642 C9O1EK 16225869 IC50 = 0.8 nM T46642 CNB43V 16226272 IC50 = 0.7 nM T46642 CIB4H9 16226487 IC50 = 1.3 nM T46642 C08URO 16226489 IC50 = 1.4 nM T46642 CO34AJ 16433103 IC50 = 6000 nM T46642 CLIM80 16996305 IC50 > 10000 nM T46642 C7PFS2 18947532 IC50 = 428 nM T46642 C64RDE 18947567 IC50 = 85 nM T46642 C7BS9F 18947582 IC50 = 2.8 nM T46642 CE20DX 18947611 IC50 = 27 nM T46642 CNRQ45 18947631 IC50 = 1955 nM T46642 CA9OG4 19010876 IC50 = 350 nM T46642 CW4BC3 19097504 IC50 = 3 nM T46642 CLR0Q2 19098329 IC50 = 59 nM T46642 CW6EM0 19098336 IC50 = 48 nM T46642 CBR1H2 19098341 IC50 = 70 nM T46642 CA0HV1 19098343 IC50 = 8 nM T46642 C3ZU8T 19108526 IC50 = 2 nM T46642 CDE7J4 19789803 IC50 = 14 nM T46642 CLS5X8 21847229 IC50 = 387 nM T46642 C4KG8A 44278976 IC50 = 4 nM T46642 CJH74Q 44286167 IC50 = 2 nM T46642 CDX93K 44316720 IC50 = 8 nM T46642 CAZN47 44316788 IC50 = 8 nM T46642 CA61TI 44316792 IC50 = 13 nM T46642 CE6SY3 44316911 IC50 = 26 nM T46642 CCOB96 44316959 IC50 = 48 nM T46642 C65LXH 44316960 IC50 = 16 nM T46642 C3VRG5 44316984 IC50 = 11 nM T46642 C46BDT 44317055 IC50 = 5 nM T46642 CQA6X4 44317063 IC50 = 40 nM T46642 CQO01T 44317064 IC50 = 73 nM T46642 CO31RQ 44317065 IC50 = 186 nM T46642 C4CI9Z 44317126 IC50 = 62 nM T46642 CI3BM4 44390722 IC50 > 1000 nM T46642 CR9Y0Z 44447696 IC50 = 145 nM T46642 CQJ85I 44447697 IC50 = 127 nM T46642 CY46GC 44447698 IC50 = 182 nM T46642 C8VCY0 44447699 IC50 = 98 nM T46642 CFI17Z 44447700 IC50 = 2070 nM T46642 C1O3TA 44447701 IC50 = 13.2 nM T46642 CMVU38 44447702 IC50 = 5 nM T46642 C5VG8X 44447703 IC50 = 94 nM T46642 CHF41Z 44447704 IC50 = 14 nM T46642 C6X4FV 44447705 IC50 = 3155 nM T46642 CML63C 44447706 IC50 = 3.7 nM T46642 CW3M6F 44447707 IC50 = 3.5 nM T46642 COVD23 44447708 IC50 = 8.6 nM T46642 C95PGW 44447709 IC50 = 6 nM T46642 C86VOX 44447710 IC50 = 8.6 nM T46642 CKPT39 44447711 IC50 = 6.5 nM T46642 C9BW6H 44447712 IC50 = 5.5 nM T46642 CCAM45 44447713 IC50 = 4.1 nM T46642 C4NYM8 44447714 IC50 = 18.3 nM T46642 CBQH74 44447715 IC50 = 134 nM T46642 CW2AF9 44447716 IC50 = 181 nM T46642 C24YFU 44447717 IC50 = 4.9 nM T46642 C7Q3ZH 44447718 IC50 = 7.6 nM T46642 CH93ZR 44447719 IC50 = 5.6 nM T46642 C6Z3TH 44447720 IC50 = 12.4 nM T46642 CG38UT 44447721 IC50 = 980 nM T46642 CY3P4U 44447722 IC50 = 776 nM T46642 CDO3H2 44447723 IC50 = 3595 nM T46642 CJOD60 44447724 IC50 = 22 nM T46642 CL4K9F 44447725 IC50 = 9.3 nM T46642 CP9VW5 44447726 IC50 = 4.5 nM T46642 C3FVK8 44447728 IC50 = 2.4 nM T46642 C2VZK0 44447729 IC50 = 3.7 nM T46642 CAN97B 44447730 IC50 = 4.2 nM T46642 CI37VD 44474262 IC50 = 5.5 nM T46642 CSEP-41 44474263 IC50 = 7.3 nM T46642 CB1IL2 44475193 IC50 = 7.7 nM T46642 C06OBS 44475194 IC50 = 27 nM T46642 CM37YN 44475195 IC50 = 6.5 nM T46642 CSBL94 44475353 IC50 = 6.8 nM T46642 CZEK01 44538088 IC50 = 4.6 nM T46642 C78MAO 44538089 IC50 = 8.3 nM T46642 CNXH68 44538090 IC50 = 559 nM T46642 C2TVE6 45263678 IC50 = 2.5 nM T46642 CF7L1T 45265994 IC50 = 2.4 nM T46642 CUV41F 45272765 IC50 = 205 nM T46642 CB9S3K 45273712 IC50 = 793 nM T46642 CSW5J6 46227656 IC50 > 10000 nM T46642 C7EH1J 46227657 IC50 = 19 nM T46642 C9XYL5 46227658 IC50 = 35 nM T46642 CE6U4N 46227659 IC50 > 10000 nM T46642 CRW03I 46227660 IC50 = 19 nM T46642 CF0AW4 46227661 IC50 = 581 nM T46642 CE29CJ 46227662 IC50 = 218 nM T46642 C12OSB 46227663 IC50 = 20.6 nM T46642 C7V6HM 46227664 IC50 = 1100 nM T46642 C4EOF9 46227665 IC50 = 4 nM T46642 C4YJ3D 46227666 IC50 = 441 nM T46642 C1R6XH 46227668 IC50 = 85 nM T46642 CCA19N 46227669 IC50 = 1.4 nM T46642 C2RDP9 46227670 IC50 = 50 nM T46642 CFE4I5 46227671 IC50 = 186 nM T46642 CC5TH8 46227672 IC50 = 1345 nM T46642 C8QJ3O 46227673 IC50 = 13 nM T46642 CTN8L7 46227674 IC50 = 38 nM T46642 CCD0U9 46227675 IC50 = 1805 nM T46642 CYS90C 46227676 IC50 = 616 nM T46642 C8JN2M 46227677 IC50 > 10000 nM T46642 C6CYN3 46227683 IC50 = 6 nM T46642 CGJ4S2 46227684 IC50 = 1114 nM T46642 CIN7K8 46227685 IC50 = 15.2 nM T46642 C3JP7W 46227686 IC50 = 4.7 nM T46642 CE93RW 46227687 IC50 = 74 nM T46642 C9NO8V 46227689 IC50 = 4.5 nM T46642 C41KVZ 46227690 IC50 = 1.7 nM T46642 C9GFQ5 46227691 IC50 = 2.5 nM T46642 C9E4SA 46227692 IC50 = 9.3 nM T46642 C1AN2R 46227693 IC50 = 3.8 nM T46642 C8PZU1 46235580 IC50 = 81 nM T46642 CE9CY1 46701619 IC50 = 0.5 nM T46642 C4O0QK 49821278 IC50 > 20000 nM T46642 C2GS8I 56837376 IC50 = 140 nM T46642 CC2BT3 56837589 IC50 > 1000 nM T46642 CH2AY6 56838673 IC50 = 2.1 nM T46642 C3OE8N 56838888 IC50 = 14 nM T46642 C3ZYO2 56839757 IC50 = 30 nM T46642 C1GR8B 56840400 IC50 = 370 nM T46642 CPZF54 56848512 IC50 = 1.9 nM T46642 CBX50A 56848641 IC50 = 2.4 nM T46642 CX05UK 56848643 IC50 = 400 nM T46642 CFU08N 56848702 IC50 = 8.3 nM T46642 C4VOX2 56848704 IC50 = 440 nM T46642 CSL04N 56848706 IC50 = 340 nM T46642 CRIM78 56848769 IC50 = 2100 nM T46642 CEZ3D0 56848825 IC50 = 2.4 nM T46642 CS4HV0 56848883 IC50 = 5.7 nM T46642 CV47AT 56848941 IC50 = 8.1 nM T46642 CB6JR7 56848995 IC50 = 1 nM T46642 CP56QN 56849238 IC50 = 100 nM T46642 C0SV7W 56849428 IC50 = 18 nM T46642 C9CI5F 56849429 IC50 = 36 nM T46642 CR85DQ 56849697 IC50 = 22.6 nM T46642 CD93FH 56849699 IC50 = 456 nM T46642 C1OYZ0 56849700 IC50 = 3220 nM T46642 CM9G8Q 56849840 IC50 = 1.7 nM T46642 CV8H2E 56849841 IC50 = 1.4 nM T46642 CV4HD0 56849842 IC50 = 1250 nM T46642 CS21JD 56849843 IC50 = 1.1 nM T46642 C18GRU 56849971 IC50 = 21.8 nM T46642 C2V3YW 56849972 IC50 = 0.5 nM T46642 C2ME6N 56849973 IC50 = 0.6 nM T46642 CR43DO 56849974 IC50 = 0.7 nM T46642 CJK39Q 56850116 IC50 = 0.7 nM T46642 C4P9FJ 56850117 IC50 = 229 nM T46642 CT92YV 56850118 IC50 = 208 nM T46642 CFND85 56850119 IC50 = 114 nM T46642 C7GZX6 56850252 IC50 = 26.8 nM T46642 CJRD42 56850253 IC50 = 19.7 nM T46642 CLS18K 56850254 IC50 = 0.8 nM T46642 CC73ZT 56850255 IC50 = 2.1 nM T46642 CA1K4C 56850391 IC50 = 0.4 nM T46642 CJ73XD 56850393 IC50 = 1.5 nM T46642 CQ9HO1 56850394 IC50 = 32600 nM T46642 CM03XK 56850522 IC50 = 0.5 nM T46642 C2XBJ9 56850523 IC50 = 1.4 nM T46642 CUY28J 56850524 IC50 = 2.2 nM T46642 CK0I6Q 56850525 IC50 = 0.4 nM T46642 CLJA61 56850666 IC50 = 0.6 nM T46642 C17IMA 56850667 IC50 = 0.5 nM T46642 C4ZS8Q 56850668 IC50 = 0.6 nM T46642 C0BM5L 56944031 IC50 = 280 nM T46642 CX1J7F 56944231 IC50 = 17 nM T46642 CO3BJ9 56944323 IC50 = 33 nM T46642 CZV5N7 56944712 IC50 = 28 nM T46642 CXK09Y 56944713 IC50 = 13 nM T46642 CV96DB 56944901 IC50 = 8.8 nM T46642 CHY3O9 56945090 IC50 = 164 nM T46642 CK87XJ 56952040 IC50 = 54 nM T46642 CLT76Y 56952460 IC50 = 23 nM T46642 C28AQB 56952861 IC50 = 1.5 nM T46642 CQN90W 56952953 IC50 = 16 nM T46642 CRU24I 56952955 IC50 = 41 nM T46642 C5FO4D 56952957 IC50 = 2.9 nM T46642 CLA05I 56953338 IC50 = 6.3 nM T46642 C9OBP3 56953432 IC50 = 19 nM T46642 CVO1U5 56953526 IC50 = 6.6 nM T46642 CG87XJ 57813859 IC50 = 3.2 nM T46642 CV9NS7 57911914 IC50 = 96 nM T46642 CWM6A0 60168044 IC50 = 240 nM T46642 CH97TU 66560743 IC50 = 1.9 nM T46642 CFOT53 66560996 IC50 = 120 nM T46642 CYC4J5 66561075 IC50 = 190 nM T46642 CCAY82 66561076 IC50 = 180 nM T46642 CK6H2U 66561077 IC50 = 160 nM T46642 CKN2U0 66764813 IC50 = 1.7 nM T46642 CA0H8X 66765152 IC50 = 1.6 nM T46642 CG90DF 66765153 IC50 = 7.7 nM T46642 CW1KQ8 66765267 IC50 = 1.1 nM T46642 C39GVZ 66765453 IC50 = 55 nM T46642 C4RJW6 66780087 IC50 = 21 nM T46642 CO1GX8 66780249 IC50 = 3.7 nM T46642 CND57Z 66780354 IC50 = 2.6 nM T46642 CVR03T 66780496 IC50 = 11 nM T46642 CRDW19 66824690 IC50 = 18 nM T46642 C19AMY 66825847 IC50 = 173 nM T46642 C57BIH 66825947 IC50 = 92 nM T46642 C6IU5J 66828210 IC50 = 14 nM T46642 CW01OL 66828211 IC50 = 14 nM T46642 CN7WR0 66828259 IC50 = 13 nM T46642 CPBG42 66828295 IC50 = 81 nM T46642 CX5P0T 66828300 IC50 = 43 nM T46642 C27KFP 66828416 IC50 = 3 nM T46642 CS57OQ 68049848 IC50 = 2.6 nM T46642 CQ50YV 68049858 IC50 = 21 nM T46642 CK6QF7 68049924 IC50 = 5.2 nM T46642 CI6KX0 68049926 IC50 = 15 nM T46642 CX5Y4U 68050144 IC50 = 2 nM T46642 CIH85M 68050153 IC50 = 18 nM T46642 CLW24G 68050156 IC50 = 1.2 nM T46642 C13HTY 68050181 IC50 = 6.7 nM T46642 CKZ1Q7 68050692 IC50 = 190 nM T46642 CLR0Q3 68074900 IC50 = 340 nM T46642 C4E6XS 68074901 IC50 = 6.2 nM T46642 C9FZ4H 68074929 IC50 = 2.2 nM T46642 C3D8AV 68074931 IC50 = 1.4 nM T46642 C02LWX 68074963 IC50 = 3.6 nM T46642 C3OIP2 68074990 IC50 = 3.6 nM T46642 C76PQD 68074998 IC50 = 2.4 nM T46642 C4P6CL 68075031 IC50 = 13 nM T46642 C6C3ZH 68075035 IC50 = 14 nM T46642 CGW5L9 68075088 IC50 = 3.5 nM T46642 CWKG52 68075192 IC50 = 160 nM T46642 CT8VP4 68075206 IC50 = 6.5 nM T46642 C08HFD 68075211 IC50 = 4 nM T46642 CS9Q1R 68075361 IC50 = 1.9 nM T46642 CA9W3J 68075551 IC50 = 18 nM T46642 CP9HB5 68075554 IC50 = 35 nM T46642 C8RY5S 68183009 IC50 = 324 nM T46642 CE91ZK 68893091 IC50 = 5.2 nM T46642 CS7MD3 68999789 IC50 = 3.6 nM T46642 CWOV98 70681615 IC50 = 2.3 nM T46642 CXBQ31 70681616 IC50 = 20 nM T46642 CDJ3I4 70681633 IC50 = 5 nM T46642 CB5S7K 70681749 IC50 > 10000 nM T46642 CGXW39 70681750 IC50 = 4500 nM T46642 CY2IB6 70681751 IC50 = 1950 nM T46642 CZ51IG 70681753 IC50 > 10000 nM T46642 CEK0D6 70683734 IC50 = 9.5 nM T46642 CW49KB 70683735 IC50 = 2.5 nM T46642 CH14PA 70683736 IC50 = 5.5 nM T46642 CYAX78 70683737 IC50 = 15 nM T46642 CKD0Z9 70683738 IC50 = 6.3 nM T46642 C4YG0A 70683756 IC50 = 1.1 nM T46642 C15IVT 70683757 IC50 = 2.9 nM T46642 CNH4M1 70683858 IC50 = 250 nM T46642 CZYQ53 70683859 IC50 = 4000 nM T46642 C9DPR4 70683863 IC50 = 2800 nM T46642 C62WLE 70685883 IC50 = 5.5 nM T46642 CZR2Y8 70685884 IC50 = 58 nM T46642 C3GV2D 70685885 IC50 = 5.8 nM T46642 CW8XH0 70685902 IC50 = 2.2 nM T46642 CT39BC 70685903 IC50 = 2.5 nM T46642 C7C6OS 70685904 IC50 = 2.4 nM T46642 CG3Q6M 70685997 IC50 = 4400 nM T46642 C7XR1H 70685998 IC50 > 10000 nM T46642 CVG8U1 70686003 IC50 = 500 nM T46642 CYW4C5 70688009 IC50 = 1315 nM T46642 CKM56W 70688010 IC50 = 2304 nM T46642 CZD25F 70688025 IC50 = 189 nM T46642 C8FQN1 70688026 IC50 = 2.9 nM T46642 C7DA9M 70688027 IC50 = 2.4 nM T46642 CD3LT1 70688028 IC50 = 1.7 nM T46642 CXE6C3 70688122 IC50 = 2500 nM T46642 CJ4Y3B 70688123 IC50 > 10000 nM T46642 CKIB98 70688128 IC50 = 3000 nM T46642 C9WED2 70690035 IC50 = 7.4 nM T46642 C13NFC 70690036 IC50 = 16 nM T46642 CP49XG 70690037 IC50 = 50 nM T46642 CQX03D 70690058 IC50 = 2.8 nM T46642 CMO6N7 70690155 IC50 = 2300 nM T46642 C5K8OC 70690156 IC50 = 250 nM T46642 CV4CM0 70690158 IC50 = 2800 nM T46642 C5FW4R 70692191 IC50 = 5.6 nM T46642 C9FZO4 70692315 IC50 = 4900 nM T46642 C0I7RU 70692316 IC50 = 450 nM T46642 CZ5Q1R 70692317 IC50 = 6000 nM T46642 CBZC10 70692318 IC50 = 700 nM T46642 C6VB5I 70694253 IC50 = 2.1 nM T46642 CA1H8L 70694254 IC50 = 3700 nM T46642 CK7B2N 70694270 IC50 = 0.8 nM T46642 C20PJR 70694271 IC50 = 1.1 nM T46642 CT6A9M 70694373 IC50 > 10000 nM T46642 CK05ND 70694374 IC50 = 9400 nM T46642 CFQ3Y5 70696344 IC50 = 4 nM T46642 CD2R5C 70696345 IC50 = 3 nM T46642 CD8M6C 70696346 IC50 = 48 nM T46642 C1CJ6M 70696347 IC50 = 7.1 nM T46642 CQX2R6 70696362 IC50 = 5.4 nM T46642 CB1N8L 70696363 IC50 = 2.6 nM T46642 CMQ17I 70696451 IC50 > 10000 nM T46642 C8X5TN 70696452 IC50 = 5000 nM T46642 CUX89H 70696453 IC50 > 10000 nM T46642 C6N9OA 70696454 IC50 = 10000 nM T46642 CH7X1Q 70696456 IC50 > 10000 nM T46642 C6UNW9 70696457 IC50 = 830 nM T46642 C68SZK 71449152 IC50 = 6 nM T46642 C2LPM4 101038239 IC50 = 12 nM T46642 C4QA9X 118536041 IC50 = 4100 nM T46642 CAG8I9 118536042 IC50 = 1700 nM T46642 C6JPZ0 118536045 IC50 = 1400 nM T46642 CTV45Z 118536050 IC50 = 1300 nM T46642 CO78DP 118536053 IC50 = 1200 nM T46642 C7HEO0 118536059 IC50 = 4100 nM T46642 CCVQ08 118536062 IC50 > 10000 nM T46642 COVA12 118536071 IC50 = 770 nM T46642 C34YNU 118734856 IC50 > 1000 nM T46642 CXP73N 122678088 IC50 = 36 nM T46642 C6MHT7 122678138 IC50 = 35 nM T46642 C4PO8H 122678183 IC50 = 29 nM T46642 C2O5TA 122678189 IC50 = 24 nM T46642 C1YK2E 122678192 IC50 = 34 nM T46642 CJI0V2 124189308 IC50 = 31.62 nM T46642 CN6S5Z 127032928 IC50 = 240 nM T46642 CVP89K 134133510 IC50 = 150 nM T46642 CLG60K 134141312 IC50 = 170 nM T46642 C9JY5N 134144042 IC50 = 26 nM T46642 C3OGS5 134145354 IC50 = 210 nM T46642 C1FW8B 134157461 IC50 = 120 nM T46642 C2RZN8 135305974 IC50 = 19.95 nM T46642 C9IH2B 135601507 IC50 = 4400 nM T46642 C5AZJ9 135651710 IC50 = 9100 nM T46642 C0VU2B 136074282 IC50 = 2.3 nM T46642 CL08BP 136074283 IC50 = 2.5 nM T46642 C3UH2X 136074284 IC50 = 2.9 nM T46642 C8GZW6 137631796 IC50 = 53 nM T46642 CN0WI4 137634303 IC50 = 92 nM T46642 CHST47 137636980 IC50 = 12 nM T46642 C3EKA0 137639989 IC50 = 46 nM T46642 C9BD1K 137642383 IC50 = 11 nM T46642 CZN23U 137642724 IC50 = 16 nM T46642 CAQ78C 137642758 IC50 = 160 nM T46642 C6SVF0 137647618 IC50 = 1 nM T46642 C71ITE 137652384 IC50 = 17 nM T46642 CAD7V8 137653372 IC50 = 29 nM T46642 CI7UG2 137657524 IC50 = 5.6 nM T46642 CT9RL1 137659038 IC50 = 115 nM T46642 CBH31L 137659953 IC50 = 324 nM T46642 CZ1Y2U 137661557 IC50 = 48 nM T46642 CHP08L 145982760 IC50 = 420 nM T46642 C9VL0R 145982804 IC50 > 10000 nM T46642 C98TPG 145982895 IC50 = 370 nM T46642 CAV47D 145982991 IC50 = 200 nM T46642 CQ1N4P 145982995 IC50 = 280 nM T46642 CHO62M 145983019 IC50 = 1700 nM T46642 CGLU58 145983160 IC50 = 74 nM T46642 CRV8O5 145983337 IC50 = 180 nM T46642 C9DM3B 145983346 IC50 = 100 nM T46642 CS8KA1 145983375 IC50 = 450 nM T46642 CQB5W4 145983395 IC50 = 150 nM T46642 C5R4DF 145983586 IC50 = 180 nM T46642 CW2L6G 145983594 IC50 = 260 nM T46642 CU95NM 145983649 IC50 = 50 nM T46642 C40IAE 145983878 IC50 = 400 nM T46642 C1HA6R 145984213 IC50 = 370 nM T46642 CP36ZU 145984302 IC50 = 190 nM T46642 CP7S4O 145984322 IC50 = 3800 nM T46642 CRTB67 145984745 IC50 = 270 nM T46642 CFW1E3 145984768 IC50 = 8800 nM T46642 C3O4TM 145984813 IC50 = 90 nM T46642 CHW74N 145984975 IC50 = 700 nM T46642 CO6I7V 145984976 IC50 = 1100 nM T46642 C5BS1R 145985135 IC50 = 18000 nM T46642 C76ACJ 145985137 IC50 = 50 nM T46642 C1UB2I 145985235 IC50 = 130 nM T46642 CM62SF 145985303 IC50 = 40 nM T46642 CBY71H 145985815 IC50 = 250 nM T46642 C6A9KY 145985817 IC50 = 320 nM T46642 CV3O6S 145985963 IC50 = 660 nM T46642 C9CTA8 145985990 IC50 = 160 nM T46642 C6T4WX 145986003 IC50 > 1000 nM T46642 C8L1FT 145986249 IC50 = 280 nM T46642 C1PV3S 145991165 IC50 = 4400 nM T46642 C6N8JT 155510634 IC50 = 101 nM T46642 C9KPR8 155515512 IC50 = 316.23 nM T46642 CDP7E5 155516065 IC50 = 100 nM T46642 CBF7H9 155516998 IC50 = 1000 nM T46642 C28CBX 155519668 IC50 = 241 nM T46642 C6QJ8R 155524126 IC50 = 251.19 nM T46642 C1FUR4 155525505 IC50 = 10 nM T46642 CV3H9Y 155526726 IC50 = 63.1 nM T46642 CW5TM8 155529670 IC50 = 25.12 nM T46642 C2QB7A 155534427 IC50 = 12.59 nM T46642 C1M9LZ 155535185 IC50 = 15.85 nM T46642 CX7PM4 155535638 IC50 = 199.53 nM T46642 C3F8NR 155536006 IC50 = 63.1 nM T46642 C8HQ0J 155537060 IC50 = 47 nM T46642 CRG48A 155540219 IC50 = 251.19 nM T46642 CWKC38 155542504 IC50 = 7943.28 nM T46642 CCRP96 155543235 IC50 = 2511.89 nM T46642 CCT43Y 155543308 IC50 = 1000 nM T46642 C41KYX 155544125 IC50 = 1000 nM T46642 C57ICR 155544322 IC50 = 12.59 nM T46642 C8WGH1 155544876 IC50 = 15.85 nM T46642 CND38C 155545031 IC50 = 59 nM T46642 CV13XI 155546721 IC50 = 39.81 nM T46642 CRN8Z6 155547317 IC50 = 31.62 nM T46642 CT46FY 155552934 IC50 = 501.19 nM T46642 COK95C 155555928 IC50 = 63.1 nM T46642 CRA05Z 155555980 IC50 = 50.12 nM T46642 C2OJS0 155558755 IC50 = 125.89 nM T46642 CKZT21 155559364 IC50 = 5.8 nM T46642 C9WYD3 155560536 IC50 = 17 nM T46642 C0RT6V 155562917 IC50 = 25118.86 nM T46642 CD51RB 155564602 IC50 = 794.33 nM T46642 CS47JC 155567408 IC50 = 63.1 nM T46642 D03NMM 46843035 IC50 = 2 nM T46642 D05FKT 9960281 IC50 = 22000 nM T46642 D0YW6B 44627267 IC50 = 2.2 nM T35734 D03RTS 2662 IC50 > 1000 nM T35734 D05ATI 3423265 IC50 = 5500 nM T35734 D05DVP 5717 IC50 = 2000 nM T35734 D05VLS 5090 IC50 > 1000 nM T35734 D09GDD 11167602 IC50 = 0.5 nM T35734 D09JUG 60490 IC50 = 591 nM T35734 D0JO7Y 104741 IC50 = 6 nM T35734 D0K8KX 5280343 IC50 = 33540 nM T35734 D0M9DC 4614 IC50 = 70000 nM T35734 D0R0MW 5329102 IC50 > 10000 nM T35734 D0R1RS 3715 IC50 > 1000 nM T35734 D0W5HK 216239 IC50 = 12 nM T35734 D04PBH 5280804 IC50 = 28430 nM T35734 D0A8KQ 59448236 IC50 = 0.028 nM T35734 D0B1FE 3194 IC50 = 110 nM T35734 D0KL3U 12000797 IC50 = 7 nM T35734 D0T5PO 5092 IC50 > 100000 nM T35734 D0U7OU 3220 IC50 = 36400 nM T35734 CZ03SB 7547 IC50 = 13 nM T35734 CS3ET7 10887 IC50 > 100000 nM T35734 CKR3L9 12116 IC50 = 70000 nM T35734 C9PH8B 14989 Ki = 27800 nM T35734 CSE1C2 19756 IC50 = 207000 nM T35734 CORX45 74805 IC50 = 1350 nM T35734 CHSZ93 75901 IC50 > 100000 nM T35734 C02SIO 95783 IC50 = 28.1 nM T35734 CVS56B 139132 IC50 = 206400 nM T35734 C0WYB1 146084 IC50 = 1370 nM T35734 C6GNU9 155380 IC50 = 26400 nM T35734 CW5Q8O 155381 IC50 = 26300 nM T35734 CHCK53 225533 IC50 = 11000 nM T35734 C92FXK 247635 IC50 = 91000 nM T35734 C46LHW 292812 IC50 = 1.7 nM T35734 CXM5V4 294966 IC50 = 8.7 nM T35734 CTH19L 442725 IC50 = 33000 nM T35734 CX1VP4 442761 IC50 = 24300 nM T35734 CD1F2K 442762 IC50 = 40600 nM T35734 CIJ6O2 471531 IC50 = 36140 nM T35734 CAI8N5 472928 IC50 = 15 nM T35734 CEM5X2 503733 IC50 = 37500 nM T35734 C30FYJ 563453 IC50 > 10000 nM T35734 CPN65F 617555 IC50 > 10000 nM T35734 CUX7D0 644455 IC50 = 1600 nM T35734 CB8QO2 644639 IC50 = 34810 nM T35734 CHV8Z1 651455 IC50 = 1498 nM T35734 CRZB53 669716 IC50 = 280 nM T35734 CD7LE4 680672 IC50 = 21000 nM T35734 C8YQ6J 689104 IC50 = 49600 nM T35734 CL81FT 694963 IC50 = 75000 nM T35734 C15EQU 727750 IC50 = 70000 nM T35734 C1S4ER 744225 IC50 = 18000 nM T35734 CLH3G2 759495 IC50 = 61000 nM T35734 C15EBP 801692 IC50 = 1400 nM T35734 CN40MG 804288 IC50 = 950 nM T35734 CLF10V 828288 IC50 = 5500 nM T35734 C0RP8F 839616 IC50 = 251 nM T35734 C4MT1H 871502 IC50 = 91000 nM T35734 C57TZF 893568 IC50 = 470 nM T35734 C09JDB 924716 IC50 = 3500 nM T35734 CLCG81 938024 IC50 = 133000 nM T35734 CQX7D3 980457 IC50 = 15.8 nM T35734 COFZ07 1004010 IC50 = 590 nM T35734 C9NQZ1 1072839 IC50 = 1200 nM T35734 C4Y6GQ 1075447 IC50 = 450 nM T35734 CGJ97Z 1088329 IC50 = 360 nM T35734 CM6SK3 1090888 IC50 = 37.3 nM T35734 CCL65Z 1090889 IC50 = 16.4 nM T35734 CR0U5L 1220478 IC50 = 379000 nM T35734 CG30IP 1276475 IC50 = 560 nM T35734 CYID94 1306384 IC50 = 20 nM T35734 C4MQ0N 1326327 IC50 = 570 nM T35734 CN0W4A 1327626 IC50 = 510 nM T35734 CLA78P 1817785 IC50 = 9000 nM T35734 CH1NL6 1845020 IC50 = 18 nM T35734 C1YVK3 2053793 IC50 = 870 nM T35734 CY2G9Z 2059107 IC50 = 1900 nM T35734 COFZ78 2061174 IC50 > 500000 nM T35734 C6G0FZ 2110176 IC50 = 7.9 nM T35734 C3F1UR 2111376 IC50 = 200 nM T35734 CQ0PF6 2133297 IC50 = 84.4 nM T35734 CJ97SP 2207161 IC50 = 25.1 nM T35734 C5OGK6 2298971 IC50 = 3000 nM T35734 CG36KX 2497562 IC50 = 29000 nM T35734 CZPW64 2666601 IC50 = 15000 nM T35734 C8J9WI 2735955 IC50 = 49000 nM T35734 C2NY0D 2764076 IC50 = 150000 nM T35734 CSZW49 2777786 IC50 = 1200000 nM T35734 C81MYO 2783031 IC50 = 52000 nM T35734 CW8LI4 2813415 IC50 = 171000 nM T35734 C9OVD4 2820615 IC50 = 9.6 nM T35734 CT5K2W 2831687 IC50 = 11.2 nM T35734 CJ25QG 2863446 IC50 = 63.7 nM T35734 C07KHU 2864086 IC50 = 610.4 nM T35734 CT3D2R 2874455 IC50 = 12828 nM T35734 CZON23 2921482 IC50 = 510 nM T35734 CZ06JK 2945280 IC50 = 234 nM T35734 C1WYZ3 2956683 IC50 = 0.5 nM T35734 CPBN09 2966629 IC50 = 6300 nM T35734 CD02CT 2982952 IC50 = 1 nM T35734 CDP03E 3010155 IC50 = 1.2 nM T35734 CPIE54 3107848 IC50 = 2680 nM T35734 C45BHQ 3115361 IC50 = 3200 nM T35734 CJ0U5T 3411092 IC50 = 34.7 nM T35734 CYX08N 3496707 IC50 = 8.2 nM T35734 C51UJQ 3575503 IC50 = 260 nM T35734 CI9ZM1 3754047 IC50 = 0.4 nM T35734 C0X3WL 3758167 IC50 = 16 nM T35734 CKZ19U 3759481 IC50 = 1800 nM T35734 C8T6BC 3776055 IC50 = 61.4 nM T35734 C2AL1X 3798558 IC50 > 100000 nM T35734 CP74IR 3826889 IC50 > 1000 nM T35734 C3AB2K 4009612 IC50 = 14 nM T35734 C5GES8 4050954 IC50 = 710 nM T35734 CGK8E3 4063047 IC50 = 6200 nM T35734 CJ7TW4 4183634 IC50 > 10000 nM T35734 CLDW53 4199500 IC50 = 1130 nM T35734 C9E6ZT 4231179 IC50 = 1.8 nM T35734 C4EH7Z 4450442 IC50 = 27.4 nM T35734 C46FDC 4460996 IC50 = 580000 nM T35734 CGY24T 4463317 IC50 = 195000 nM T35734 C8VPI0 4465413 IC50 = 0.4 nM T35734 C1RQ8S 4519806 IC50 = 250 nM T35734 CX17FN 4550519 IC50 > 100000 nM T35734 CZ9E1B 4560409 IC50 = 23 nM T35734 CQX9J2 4626092 IC50 = 1048 nM T35734 C4IM1E 4686891 IC50 = 83 nM T35734 C7V2TK 4799088 IC50 = 0.8 nM T35734 C9HJ3X 4805349 IC50 = 1100 nM T35734 C2L5EW 5048923 IC50 = 2.4 nM T35734 CB9F5Q 5053944 IC50 = 551 nM T35734 CC5M8A 5190631 IC50 = 1224 nM T35734 CM73PF 5220350 IC50 = 430 nM T35734 CJ5P7R 5235274 IC50 = 174 nM T35734 CH50QK 5281643 IC50 = 21760 nM T35734 CRBV34 5315874 IC50 = 1100 nM T35734 C9OUN7 5317701 IC50 = 20000 nM T35734 CUD6H5 5318606 IC50 = 17230 nM T35734 C1EB3J 5319526 IC50 = 1000 nM T35734 C21EUO 5357283 IC50 = 1800 nM T35734 C3T5QA 5480249 IC50 = 18050 nM T35734 CU16IF 6438381 IC50 = 2040 nM T35734 CSA24L 6474310 IC50 = 2800 nM T35734 CB6R8N 7017351 IC50 = 800000 nM T35734 CD6I1H 7060576 IC50 = 2200000 nM T35734 CLD97X 7545432 IC50 = 400 nM T35734 C1U9CK 7546299 IC50 = 8.1 nM T35734 C71HEJ 8744203 IC50 = 159 nM T35734 C9JKH4 9082162 IC50 = 2100 nM T35734 CD3VJ1 9166073 IC50 = 100 nM T35734 CT3MG6 9217979 IC50 = 34 nM T35734 CHB36V 9820664 IC50 = 41 nM T35734 CL73SJ 9866696 IC50 = 37400 nM T35734 CA08ES 10031482 IC50 = 18640 nM T35734 CXF09G 10072550 IC50 = 2 nM T35734 C52TFA 10358670 IC50 = 5.1 nM T35734 C5FQ2C 10754392 IC50 = 3260 nM T35734 CL1IQ3 10989222 IC50 = 2.6 nM T35734 CEJR28 11020253 IC50 = 358000 nM T35734 C3V0OK 11020645 IC50 = 78000 nM T35734 CPKS64 11053022 IC50 = 70000 nM T35734 C6I7PV 11185623 IC50 = 1020 nM T35734 C93TFX 11186401 IC50 = 2100 nM T35734 CE2U6G 11186477 IC50 > 100000 nM T35734 C3KSL1 11186504 IC50 = 22000 nM T35734 CW5S0Q 11187224 IC50 = 10 nM T35734 CTXF95 11198157 IC50 = 5000 nM T35734 C3Y1DN 11200931 IC50 = 110 nM T35734 C4NX9M 11209573 IC50 = 5900 nM T35734 C3TK0O 11211985 IC50 = 130 nM T35734 C7O0TC 11212321 IC50 = 1.6 nM T35734 CP2I8M 11212905 IC50 = 140 nM T35734 CW01ZJ 11223497 IC50 = 2.3 nM T35734 CO7CZ5 11236241 IC50 = 0.8 nM T35734 C63SGL 11247888 IC50 = 1.3 nM T35734 C04LEI 11265133 IC50 > 100000 nM T35734 CF8N4U 11268605 IC50 = 390 nM T35734 CK3L0N 11270379 IC50 = 1.8 nM T35734 C6M3EC 11280933 IC50 = 14 nM T35734 CNYV70 11282175 IC50 = 100 nM T35734 C7DW1N 11293505 IC50 = 120 nM T35734 CE8YR0 11299717 IC50 > 10000 nM T35734 C4JZ1M 11303864 IC50 = 2 nM T35734 CYS6Q4 11305487 IC50 = 110 nM T35734 C45KMY 11329622 IC50 = 100 nM T35734 CL8V5P 11340005 IC50 = 200 nM T35734 C61LQZ 11360061 IC50 = 2400 nM T35734 C9CW3P 11362503 IC50 = 1 nM T35734 CK8A0Q 11362548 IC50 = 100 nM T35734 CZ20UB 11371517 IC50 = 430 nM T35734 CLP3O5 11373914 IC50 = 1 nM T35734 CM03CT 11379742 IC50 = 38000 nM T35734 C8FD6K 11381825 IC50 = 2100 nM T35734 C2B4FE 11381826 IC50 = 26000 nM T35734 CCX5N2 11397754 IC50 = 100 nM T35734 CX1HS8 11404645 IC50 > 100000 nM T35734 CS0GW1 11416182 IC50 = 25200 nM T35734 CH7VI2 11416405 IC50 = 9400 nM T35734 C4FLH8 11425995 IC50 = 37000 nM T35734 C0LJX5 11427381 IC50 > 100000 nM T35734 CN6S1Z 11427448 IC50 > 100000 nM T35734 C1XMF2 11431539 IC50 = 100 nM T35734 C7IS1F 11437855 IC50 = 1600 nM T35734 CQ8A2T 11441534 IC50 = 4.3 nM T35734 CY27OC 11448009 IC50 > 100000 nM T35734 CMJ90I 11472902 IC50 > 100000 nM T35734 C9WX5L 11474480 IC50 = 540 nM T35734 C1VYD3 11484196 IC50 > 100000 nM T35734 CJWT81 11484242 IC50 = 18000 nM T35734 CD6S8N 11486246 IC50 = 120 nM T35734 CC0SD7 11487324 IC50 = 2.9 nM T35734 CZNH72 11489483 IC50 = 2.4 nM T35734 CDZ0T8 11494154 IC50 = 19.9 nM T35734 CN2U7C 11494688 IC50 = 0.9 nM T35734 C9W8BT 11494940 IC50 = 10 nM T35734 CR2L4V 11502402 IC50 = 1.6 nM T35734 CS7HL4 11519728 IC50 = 55 nM T35734 C2ZF4D 11525463 IC50 = 1.7 nM T35734 C2PF8R 11532957 IC50 = 1.7 nM T35734 CZ5XW8 11546213 IC50 = 0.5 nM T35734 C31BJY 11552964 IC50 = 2.3 nM T35734 CX58GE 11553060 IC50 = 0.5 nM T35734 CM38PX 11559025 IC50 = 1.3 nM T35734 CY8N4B 11574457 IC50 = 2.5 nM T35734 C0LKE1 11581328 IC50 = 0.7 nM T35734 C2HCO7 11595336 IC50 = 126 nM T35734 CW3HD2 11596176 IC50 = 0.5 nM T35734 C7S3LH 11603291 IC50 = 4 nM T35734 CFT90C 11603817 IC50 = 0.82 nM T35734 CDQ5O2 11603833 IC50 = 90 nM T35734 C02NLP 11604843 IC50 = 1.5 nM T35734 C8PZ5F 11610101 IC50 = 1200 nM T35734 CZM5R4 11618153 IC50 = 247 nM T35734 C2WYC8 11619213 IC50 = 58 nM T35734 CMX54I 11619802 IC50 = 4.2 nM T35734 C6BKX0 11624930 IC50 = 0.8 nM T35734 C7GS9I 11631634 IC50 = 0.5 nM T35734 CFI85V 11641460 IC50 = 3.5 nM T35734 CA3O2S 11655334 IC50 = 1.4 nM T35734 CQEG95 11683650 IC50 = 57.9 nM T35734 C60DYL 11771739 IC50 = 32000 nM T35734 C18UXP 11976367 IC50 = 18 nM T35734 C8M3OT 11976769 IC50 = 5 nM T35734 CFB4R8 11976771 IC50 = 5 nM T35734 C0AIR3 12307752 IC50 = 229 nM T35734 CX9ZM4 14149310 IC50 = 19.5 nM T35734 CH62MC 14626814 IC50 = 2500 nM T35734 CKMB21 14626863 IC50 = 590 nM T35734 CL18DN 15632681 IC50 = 6800 nM T35734 C89WYZ 16038368 IC50 = 0.5 nM T35734 CJ9WX7 16041611 IC50 = 2.5 nM T35734 C71MXZ 16046139 IC50 = 1370 nM T35734 CN0B4F 16049792 Ki = 15 nM T35734 C8UKZ1 16066763 IC50 = 1.2 nM T35734 CE4DB6 16095497 IC50 = 2000 nM T35734 CT1HY4 16096935 IC50 > 10000 nM T35734 CUS7L2 16227558 IC50 = 127000 nM T35734 CES52O 16340771 IC50 = 136 nM T35734 CF39OH 16375826 IC50 = 7400 nM T35734 CV3Z5Q 16654086 IC50 = 57000 nM T35734 C52CXV 16679589 IC50 = 2.6 nM T35734 C23MQT 16725330 EC50 = 0.14 nM T35734 C26LFK 16725813 IC50 = 18 nM T35734 CN5GT7 16739030 IC50 = 5.1 nM T35734 CO9E8F 16755961 IC50 = 1.6 nM T35734 CX86BW 16756171 IC50 = 1.1 nM T35734 CMX3V4 16756172 IC50 = 0.64 nM T35734 C4UXN8 16756173 IC50 = 1.6 nM T35734 CPI68V 16756270 IC50 = 2.5 nM T35734 C9QYM3 16756274 IC50 = 7 nM T35734 CTO4G5 16756387 IC50 = 9.1 nM T35734 CAJU73 16756391 IC50 = 42 nM T35734 CV3H8R 16756506 IC50 = 1.8 nM T35734 CIE6C9 16756509 IC50 = 2.5 nM T35734 CGKQ13 16756511 IC50 = 2.6 nM T35734 C8G9AL 16756850 IC50 = 0.4 nM T35734 CO95PQ 16756959 IC50 = 2 nM T35734 C9FS2B 16757061 IC50 = 3.5 nM T35734 C6X3NL 16757353 IC50 = 1.9 nM T35734 CW7TG2 16757354 IC50 = 330 nM T35734 CEA73Y 17019024 IC50 = 92 nM T35734 CT3OU4 17170431 IC50 = 6.5 nM T35734 CPG3R4 17171886 IC50 = 10500 nM T35734 C3T1KI 17171912 IC50 = 8100 nM T35734 C15PMA 17205433 IC50 = 49 nM T35734 CT0AB3 17223607 IC50 = 1200 nM T35734 C93FCJ 17262315 IC50 = 345 nM T35734 CW6X7D 17270772 IC50 = 1084 nM T35734 C07BFS 17283358 IC50 = 15 nM T35734 C8BN5S 17298177 IC50 = 170 nM T35734 CWX3O9 17360242 IC50 = 4200 nM T35734 C4YCS7 17391208 IC50 = 25 nM T35734 C1J4ZT 17410717 IC50 = 32 nM T35734 C4QGW0 17486918 IC50 = 102 nM T35734 CG2KT4 17639891 IC50 = 570 nM T35734 CW9K5H 17748340 IC50 = 450 nM T35734 CS0RL1 17748379 IC50 = 9.9 nM T35734 CJ2F9C 18101825 IC50 = 113 nM T35734 CU1DK3 19575095 IC50 = 133 nM T35734 C73QOV 19576771 IC50 = 91000 nM T35734 C90FVQ 19651571 IC50 = 2592 nM T35734 CSN14A 19651576 IC50 = 451 nM T35734 CFC59I 20173062 IC50 = 281 nM T35734 CKX40H 21372902 IC50 = 42 nM T35734 CPMH45 21372904 IC50 = 50 nM T35734 CCOQ23 21372906 IC50 = 43.3 nM T35734 C0G1NP 21372918 IC50 = 200 nM T35734 CAD5J4 21454912 IC50 = 131 nM T35734 CRM76T 22978785 IC50 = 3.9 nM T35734 C39OME 22978787 IC50 = 1.1 nM T35734 CED1S5 23363908 IC50 = 1080 nM T35734 C64WVT 23581964 IC50 = 14.3 nM T35734 COS97Z 23581967 IC50 = 0.5 nM T35734 CM2TV7 23582678 IC50 = 4.5 nM T35734 CKB5Q3 23631477 IC50 = 10 nM T35734 C6ZUX4 23631561 IC50 = 9 nM T35734 CHR9E3 23631562 IC50 = 11 nM T35734 CD5MC7 23631653 IC50 = 1.8 nM T35734 C2P9YM 23631654 IC50 = 1.1 nM T35734 C9F7LC 23631732 IC50 = 1.3 nM T35734 CCKN39 23631735 IC50 = 11 nM T35734 CIUD83 23631821 IC50 = 23 nM T35734 CC8G2U 23631822 IC50 = 1.8 nM T35734 CI10WO 23729132 IC50 = 2 nM T35734 C0OZ1K 24132341 IC50 = 4.1 nM T35734 CO2HC6 24160013 IC50 = 6 nM T35734 CY63PV 24241093 IC50 = 5.8 nM T35734 C0L8QY 24744859 IC50 = 11 nM T35734 C7UMP4 24748090 IC50 = 15 nM T35734 C8ZAP1 24748125 IC50 = 27 nM T35734 C0JRN7 24748284 IC50 = 24 nM T35734 CQ6D4E 24748285 IC50 > 3000 nM T35734 CYI13F 24748286 IC50 > 3000 nM T35734 C9RML7 24748327 IC50 = 19 nM T35734 C26IRP 24748328 IC50 = 18 nM T35734 CPFI09 24748332 IC50 = 46 nM T35734 C8ES3F 24748333 IC50 = 110 nM T35734 CR4N6V 24748367 IC50 > 3000 nM T35734 C9Y5RA 24748400 IC50 > 3000 nM T35734 CT9ZU6 24748401 IC50 > 3000 nM T35734 CNJC98 24748402 IC50 = 200 nM T35734 C4JKA6 24748434 IC50 = 1500 nM T35734 CU4K6O 24748435 IC50 = 2900 nM T35734 CX8O1I 24748436 IC50 = 41 nM T35734 C4JC7E 24748473 IC50 = 1000 nM T35734 CT59LW 24748475 IC50 = 12 nM T35734 CC4GB1 24748513 IC50 = 15 nM T35734 C27DXT 24748515 IC50 = 150 nM T35734 CMT3R6 24748516 IC50 = 220 nM T35734 CF9D5S 24748556 EC50 = 4.2 nM T35734 CSG65M 24748557 IC50 = 230 nM T35734 C7G3RW 24748561 IC50 = 210 nM T35734 CG74QF 24748562 IC50 = 180 nM T35734 CR6QD8 24748603 EC50 = 10 nM T35734 C5ZYA1 24748652 IC50 = 12 nM T35734 CNCJ10 24748700 IC50 = 29 nM T35734 CR0D8W 24766020 IC50 = 2 nM T35734 CO3SJ8 24809976 IC50 = 100 nM T35734 CZ5T2C 24825713 EC50 = 1.7 nM T35734 CNU19Q 24849237 IC50 = 1.3 nM T35734 C9OS3X 24849238 IC50 = 1.2 nM T35734 CIZ2C7 24849239 IC50 = 1.7 nM T35734 CGD31H 24849240 IC50 = 2.1 nM T35734 CNU25X 24849906 IC50 = 3900 nM T35734 CO04FQ 24849907 IC50 = 2600 nM T35734 CW9T8I 24849908 IC50 = 610 nM T35734 CXL7U4 24849909 IC50 = 110 nM T35734 C5M8RN 24849911 IC50 = 2.6 nM T35734 C5JK9P 24871512 IC50 = 3.9 nM T35734 CWV5E8 24894561 IC50 = 3 nM T35734 CGF52Z 24894562 IC50 = 1 nM T35734 C5UBN0 24894570 IC50 = 1 nM T35734 C2W6VI 24894571 IC50 = 1 nM T35734 C5DP7I 24895838 IC50 = 3 nM T35734 C2TPN1 24895839 IC50 = 5 nM T35734 CR2V5I 24898133 Ki = 0.66 nM T35734 C7LG4P 24898341 Ki = 1.17 nM T35734 CJL98O 24899016 IC50 = 10 nM T35734 CBQN62 24899522 Ki = 0.49 nM T35734 C9NTJ6 24899523 IC50 = 3.7 nM T35734 C6G9WQ 24899524 IC50 = 11 nM T35734 CLD9N5 24945361 IC50 = 200 nM T35734 CA8ZC6 24945437 IC50 = 230 nM T35734 CI5J2R 24945438 IC50 = 235 nM T35734 CO96GK 24945440 IC50 = 47 nM T35734 CTDX89 24945518 IC50 = 11 nM T35734 CSE10H 24945519 IC50 = 9 nM T35734 CZ0QK9 24945520 IC50 = 8 nM T35734 CQ06RO 24945521 IC50 = 5 nM T35734 CAJ36R 24945522 IC50 = 14 nM T35734 C9FPY3 24945591 IC50 = 12 nM T35734 CT3JC8 24945594 IC50 = 160 nM T35734 CTE46N 24945676 IC50 = 4 nM T35734 CJ5N8B 24945677 IC50 = 7 nM T35734 CBYC97 24945680 IC50 = 4 nM T35734 CD0N4T 24945759 IC50 = 4 nM T35734 CN07HP 24945760 IC50 = 16 nM T35734 C2TX0G 24945761 IC50 = 2 nM T35734 CVG64T 24945762 IC50 = 15 nM T35734 CX0ZL3 24949412 IC50 > 10000 nM T35734 CVRL81 25014525 IC50 = 11 nM T35734 CPG41H 25014526 IC50 = 1880 nM T35734 CIK9C6 25014528 IC50 = 121 nM T35734 C03DBM 25014529 IC50 = 33 nM T35734 C2P0GC 25014530 IC50 = 1 nM T35734 COH0M5 25014611 IC50 = 550 nM T35734 CBF8S7 25014612 IC50 = 365 nM T35734 CDX84Q 25014613 IC50 = 14000 nM T35734 CPCU36 25014614 IC50 = 321 nM T35734 C5UI4B 25014695 IC50 = 5000 nM T35734 CZXW45 25014696 IC50 = 2 nM T35734 CPZR45 25014698 IC50 = 140 nM T35734 CS8RU4 25014699 IC50 = 54 nM T35734 C81EUT 25014700 IC50 = 116 nM T35734 CG28TW 25014701 IC50 = 55 nM T35734 CA5Y1U 25014773 IC50 = 43 nM T35734 C0HWR9 25014774 IC50 = 870 nM T35734 CIUF89 25014775 IC50 = 1.5 nM T35734 CSL7Q5 25014776 IC50 = 0.8 nM T35734 CV1A5O 25014777 IC50 = 8 nM T35734 COR28L 25014778 IC50 = 81 nM T35734 C7TB9I 25014859 IC50 = 4.8 nM T35734 CB9KR1 25014862 IC50 = 15 nM T35734 CDKF37 25014954 IC50 = 0.8 nM T35734 C4F9OY 25014955 IC50 = 0.8 nM T35734 CG8Z2U 25015038 IC50 = 110 nM T35734 C67ARV 25015040 IC50 = 22 nM T35734 C9A4YU 25015041 IC50 = 6.5 nM T35734 C5V7XW 25015042 IC50 = 390 nM T35734 CA16YS 25015043 IC50 = 28 nM T35734 C6C5SW 25015121 IC50 = 2.5 nM T35734 CXAK94 25015122 IC50 = 5.2 nM T35734 CD1SO3 25015124 IC50 = 5.4 nM T35734 CL3F2T 25015125 IC50 = 3.9 nM T35734 CHA43V 25015202 IC50 = 1550 nM T35734 CZO3H2 25015203 IC50 = 1040 nM T35734 CUV69O 25015204 IC50 = 40 nM T35734 CH1KZ7 25015205 IC50 = 1.3 nM T35734 CYG8P7 25015206 IC50 = 0.8 nM T35734 COSD76 25015279 IC50 = 0.8 nM T35734 CFKY10 25015280 IC50 = 13.8 nM T35734 C8M2OL 25015711 IC50 = 14 nM T35734 COIJ63 25015712 IC50 = 10000 nM T35734 CP0G9C 25036176 IC50 > 3000 nM T35734 CY5DP2 25040232 IC50 = 17 nM T35734 C5FRN7 25069498 IC50 = 185 nM T35734 COA51C 25069816 IC50 = 1.6 nM T35734 C9DF7E 25070135 IC50 = 29 nM T35734 CF12JM 25070137 IC50 = 6.4 nM T35734 CP7K5W 25073288 IC50 = 27 nM T35734 CNK6W2 25093348 IC50 = 2.8 nM T35734 C1DRW4 25093349 IC50 > 100000 nM T35734 C9CM5V 25093351 IC50 = 0.9 nM T35734 CF1ZN0 25093352 IC50 = 12 nM T35734 CF5AO8 25093353 IC50 = 2.9 nM T35734 C8RL2M 25109036 IC50 = 270 nM T35734 C7IMH3 25109171 IC50 = 310 nM T35734 CUM8N6 25109344 IC50 = 11 nM T35734 C3RGZ0 25138325 IC50 < 1 nM T35734 C4N8BX 25261287 IC50 = 1 nM T35734 CWYJ73 25261449 IC50 = 80 nM T35734 CU1Y6R 25261451 IC50 = 40 nM T35734 CL2NO1 25261454 IC50 = 1 nM T35734 C1IW5M 25261456 IC50 = 3 nM T35734 CRJ8H4 25261457 IC50 = 50 nM T35734 CV5FB3 25261927 IC50 = 20 nM T35734 C0VJ1S 26087384 IC50 = 8.3 nM T35734 C2TM7Q 26087504 IC50 = 2200 nM T35734 C5UCL0 26087805 IC50 = 640 nM T35734 CMB3L1 26098180 IC50 = 8.5 nM T35734 C2Y8PJ 26114956 IC50 = 1.1 nM T35734 CP3VA4 26123289 IC50 = 6 nM T35734 C07NQJ 26289048 IC50 = 23 nM T35734 CPX10D 26412245 IC50 = 30 nM T35734 CTHQ24 26413325 IC50 = 2.8 nM T35734 C5UK1A 26516405 IC50 = 78 nM T35734 CM0G8K 26516412 IC50 = 470 nM T35734 C1H4NF 26516455 IC50 = 62 nM T35734 C32SXE 26536772 IC50 = 0.6 nM T35734 C2EJX1 26574899 IC50 = 8.7 nM T35734 CHC8Z4 26641666 IC50 = 6.7 nM T35734 C2V3ES 26654855 IC50 = 20 nM T35734 CP3K9U 26693826 IC50 = 4.6 nM T35734 C2WQP6 26695748 IC50 = 18 nM T35734 CV52ZJ 26697387 IC50 = 5.2 nM T35734 CAK3Z2 26711757 IC50 = 224 nM T35734 CWK16S 26711777 IC50 = 1.6 nM T35734 C42LWZ 26711882 IC50 = 46.9 nM T35734 CJFX93 26908240 IC50 = 5.2 nM T35734 CN8F1C 26910619 IC50 = 1.7 nM T35734 C9VON1 26913868 IC50 = 45 nM T35734 C3P8FH 27167036 IC50 = 20 nM T35734 C8BH0K 27646854 IC50 = 340 nM T35734 CS6B3V 27646915 IC50 = 87.6 nM T35734 C8C2AI 27741071 IC50 = 64 nM T35734 C72FDZ 27870092 IC50 = 6.1 nM T35734 CZJ67B 28062065 IC50 = 1.2 nM T35734 C6RW7B 28080623 IC50 = 12 nM T35734 CZ49RH 28781778 IC50 = 100000 nM T35734 CIP8S5 29371674 IC50 = 23 nM T35734 C75DEZ 30726432 IC50 = 12.6 nM T35734 C7GW2X 30879131 IC50 = 39.6 nM T35734 CWN8R3 31031050 IC50 = 2.3 nM T35734 CV3RQ6 31899116 IC50 = 90 nM T35734 CIC5A6 32978914 IC50 = 320 nM T35734 CG4Y0A 33370309 IC50 > 10000 nM T35734 CQ4O7I 35014275 IC50 = 250 nM T35734 CL4PK3 39382334 IC50 = 3500 nM T35734 CQKJ76 41327880 IC50 = 3 nM T35734 CDAI28 42549315 IC50 = 290 nM T35734 C4P1IM 42643589 IC50 = 1 nM T35734 CX9SM6 42643591 IC50 = 5 nM T35734 C96FIN 42644084 IC50 < 1000 nM T35734 C8BI5F 42644088 IC50 = 12 nM T35734 CREJ31 42646199 IC50 = 5 nM T35734 CKZ76R 42646202 IC50 < 1000 nM T35734 C81NVM 42646450 IC50 = 59 nM T35734 CVBO78 42647178 IC50 < 1 nM T35734 C0NF8L 43873053 IC50 = 29.1 nM T35734 CU71TC 43873057 IC50 = 20.1 nM T35734 CIJ56L 44142782 Ki = 0.91 nM T35734 CO9AY2 44182947 IC50 = 160 nM T35734 CBPV86 44188851 IC50 = 80 nM T35734 CWM71O 44188852 IC50 = 40 nM T35734 CX4YL8 44232522 IC50 = 34 nM T35734 CCD57H 44234657 IC50 = 71.5 nM T35734 C3RN8F 44234658 IC50 = 1451 nM T35734 CLIP73 44234659 IC50 = 8484 nM T35734 CZ6M9E 44234661 IC50 = 2834 nM T35734 C08SNF 44234913 IC50 = 11064 nM T35734 CV21XB 44234918 IC50 = 58712 nM T35734 CN7Z1L 44235170 IC50 = 17622 nM T35734 CGT4Q9 44235176 IC50 = 13877 nM T35734 C7PN2M 44235410 IC50 = 17755 nM T35734 C7UY5F 44235863 IC50 = 18 nM T35734 CX2W8Y 44236320 IC50 = 7 nM T35734 C8LN0U 44236321 IC50 = 36 nM T35734 CK4S5Y 44236322 IC50 = 8 nM T35734 CY9KN8 44307465 IC50 = 253000 nM T35734 C21JPV 44416760 IC50 = 5 nM T35734 C9UE0R 44416761 IC50 = 8.7 nM T35734 CTC4Q0 44416789 IC50 = 6.7 nM T35734 C59EGT 44416791 IC50 = 3.3 nM T35734 C35LVR 44416809 IC50 = 6.2 nM T35734 C2H4TS 44416810 IC50 = 3.4 nM T35734 CMO0T7 44416831 IC50 = 1.8 nM T35734 CUCO53 44416832 IC50 = 4.1 nM T35734 C8G3DI 44416849 IC50 = 1.5 nM T35734 CET0D4 44416886 IC50 = 1.7 nM T35734 C9FX7E 44416903 IC50 = 1.1 nM T35734 CBA8G7 44416904 IC50 = 1.1 nM T35734 C8EZ5U 44416921 IC50 = 250 nM T35734 CNKR86 44416922 IC50 = 72 nM T35734 CJ3D8P 44416942 IC50 = 1.8 nM T35734 CI8TK3 44416943 IC50 = 3.2 nM T35734 CE08OD 44416944 IC50 = 160 nM T35734 C0AXN8 44416945 IC50 = 10 nM T35734 CJE3D7 44416960 IC50 = 7.6 nM T35734 CHP4K2 44416961 IC50 = 5.4 nM T35734 C45WNF 44416981 IC50 = 7.3 nM T35734 C82PSJ 44416982 IC50 = 9 nM T35734 CX18MQ 44417013 IC50 = 2.7 nM T35734 C4PS3Z 44417034 IC50 = 1.1 nM T35734 C7O2LJ 44417125 IC50 = 41 nM T35734 CR1BY8 44417126 IC50 = 400 nM T35734 CU48FD 44417169 IC50 = 43 nM T35734 C7AE2X 44417226 IC50 = 11.8 nM T35734 CU83PC 44417231 IC50 = 170 nM T35734 CY81AD 44418272 IC50 = 100 nM T35734 CP62JB 44418604 IC50 = 2700 nM T35734 CBYD60 44418605 IC50 > 100000 nM T35734 C0YC4B 44418616 IC50 > 100000 nM T35734 C0MT7A 44418617 IC50 > 100000 nM T35734 CJ3NT2 44418618 IC50 > 100000 nM T35734 CJF2Y7 44418619 IC50 > 100000 nM T35734 CX26NO 44418620 IC50 > 100000 nM T35734 CVOF02 44418623 IC50 > 100000 nM T35734 C8C0PX 44418624 IC50 > 100000 nM T35734 C9L2NQ 44418632 IC50 = 25000 nM T35734 C54NYF 44418633 IC50 = 24000 nM T35734 CXL7T3 44418634 IC50 > 100000 nM T35734 CE49YJ 44418637 IC50 = 30000 nM T35734 CKWE79 44418638 IC50 = 21000 nM T35734 C4YSV1 44418639 IC50 > 100000 nM T35734 C4XTK0 44418640 IC50 > 100000 nM T35734 CC8Y9J 44418643 IC50 = 17000 nM T35734 CJ9RK5 44418646 IC50 > 100000 nM T35734 CQD63E 44418647 IC50 > 100000 nM T35734 CXHZ79 44418648 IC50 > 100000 nM T35734 C46KRS 44418649 IC50 > 100000 nM T35734 CNM8W2 44418653 IC50 > 100000 nM T35734 CKP3F0 44418654 IC50 = 1000 nM T35734 CJ4U7Q 44418655 IC50 > 100000 nM T35734 C6AWU9 44418656 IC50 > 100000 nM T35734 C13YXS 44418667 IC50 = 41000 nM T35734 CC0M8N 44418688 IC50 = 260 nM T35734 C9F6NG 44418689 IC50 = 2100 nM T35734 CTH2J8 44418690 IC50 > 100000 nM T35734 C2QOI3 44418691 IC50 > 100000 nM T35734 CW5ES2 44418692 IC50 = 1500 nM T35734 C7D5YN 44418693 IC50 = 5500 nM T35734 CL78EF 44418694 IC50 = 130 nM T35734 CKPO67 44418695 IC50 = 880 nM T35734 C7CMD4 44418696 IC50 = 870 nM T35734 CTV9M5 44418697 IC50 = 100 nM T35734 CI9O3G 44418698 IC50 = 100 nM T35734 CZ3E0N 44418699 IC50 = 2400 nM T35734 CW1K7O 44418700 IC50 = 1300 nM T35734 CBQ3I7 44418701 IC50 = 230 nM T35734 CB94QF 44418702 IC50 = 100 nM T35734 C1SNY2 44418703 IC50 > 100000 nM T35734 C6JNY0 44418704 IC50 > 100000 nM T35734 C85FAH 44418705 IC50 = 41000 nM T35734 CZV05W 44418706 IC50 = 80000 nM T35734 CGD6E0 44418707 IC50 = 55000 nM T35734 C68XPZ 44419689 IC50 = 30 nM T35734 CCWI52 44419697 IC50 = 1 nM T35734 CKW1Z4 44419705 IC50 = 0.6 nM T35734 CAPS89 44419709 IC50 = 1.2 nM T35734 C3S6BH 44419713 IC50 = 940 nM T35734 C91VWX 44419715 IC50 = 50500 nM T35734 C04BTL 44419716 IC50 = 2.9 nM T35734 CGAI59 44419719 IC50 = 142 nM T35734 CIQH27 44419720 IC50 = 2 nM T35734 CX4E8Y 44419724 IC50 = 590 nM T35734 C7ZFA8 44419725 IC50 = 100 nM T35734 C3J4HQ 44422270 IC50 = 1.5 nM T35734 C24QRZ 44422271 IC50 = 2 nM T35734 CWA7C9 44422273 IC50 = 1.7 nM T35734 C3YUX8 44422278 IC50 = 2.1 nM T35734 C1A6TH 44422280 IC50 = 1.9 nM T35734 CG0FN6 44422288 IC50 = 100 nM T35734 C5RD1A 44422289 IC50 = 7.6 nM T35734 CLWV49 44422339 IC50 = 0.7 nM T35734 CFM62D 44427448 IC50 = 0.6 nM T35734 CP26BT 44427449 IC50 = 8300 nM T35734 C4I9DX 44464338 IC50 = 1.6 nM T35734 CG5I4T 44468933 IC50 = 0.7 nM T35734 C4M6CY 44469062 IC50 = 3.1 nM T35734 CVAD36 44474923 IC50 > 3000 nM T35734 CDTL21 44475061 IC50 = 5 nM T35734 CPH5M1 44475062 EC50 = 0.6 nM T35734 C52VLJ 44475063 EC50 = 0.3 nM T35734 CP42EV 44475203 EC50 = 2.8 nM T35734 C59RWP 44475364 IC50 = 5 nM T35734 C2ZI9A 44475365 IC50 = 5 nM T35734 CG0KR9 44475366 EC50 = 2.1 nM T35734 CSB0C1 44475367 EC50 = 0.3 nM T35734 C8X5CU 44475368 EC50 = 0.4 nM T35734 C5EX1K 44555473 IC50 = 1 nM T35734 C7MG0D 44582417 IC50 = 5.8 nM T35734 CK52BD 44582418 IC50 = 5.1 nM T35734 CY51RN 44582419 IC50 = 3.9 nM T35734 C7NM3T 44582420 IC50 = 11 nM T35734 C1V0DT 44582457 IC50 = 25 nM T35734 C3NT4W 44582458 IC50 = 28.7 nM T35734 C2P1QO 44582485 IC50 = 36 nM T35734 C4IN5T 44582487 IC50 = 4 nM T35734 CWN4Y0 44582488 IC50 = 2 nM T35734 CTU37P 44582512 IC50 = 3.1 nM T35734 CZPX05 44582513 IC50 = 116 nM T35734 C0PUJ4 44582514 IC50 = 12 nM T35734 CS9F0P 44582515 IC50 = 71 nM T35734 C0IP7C 44583234 IC50 < 1 nM T35734 C6HTC1 44583235 IC50 = 3 nM T35734 CZJU04 44583236 IC50 = 20 nM T35734 C3TYW0 44583237 IC50 = 8 nM T35734 CCL9R0 44583238 IC50 = 7 nM T35734 COX7F1 44583287 IC50 = 1 nM T35734 C5SI9Q 44583288 IC50 = 4 nM T35734 CFT74N 44583289 IC50 = 8 nM T35734 CC19TZ 44583290 IC50 < 1 nM T35734 C90RAV 44583349 IC50 < 1 nM T35734 CK81NJ 44583350 IC50 < 1 nM T35734 C20VTN 44583351 IC50 = 4 nM T35734 CD5U3A 44583352 IC50 = 4 nM T35734 C9G7VT 44583353 IC50 < 1 nM T35734 C6QF4O 44583354 IC50 < 1 nM T35734 C48AQR 44583355 IC50 < 1 nM T35734 CG5X0M 44583356 IC50 = 3 nM T35734 CUG9Y0 44583357 IC50 = 5 nM T35734 CL2I3M 44590227 IC50 = 185 nM T35734 CL2TC7 44590269 IC50 = 210 nM T35734 C4JH5P 44590337 IC50 = 1110 nM T35734 CZ4U7K 44590338 IC50 = 1540 nM T35734 C5P8WO 44590339 IC50 = 685 nM T35734 CX5V0G 44590744 IC50 = 88 nM T35734 CXF12H 44590792 IC50 = 93 nM T35734 CNS92A 44590793 IC50 = 15000 nM T35734 C74ATW 44590855 IC50 = 3600 nM T35734 CG0DC5 44590856 IC50 > 2000 nM T35734 C7MSV3 44590857 IC50 = 23 nM T35734 CQP4O2 44590934 IC50 = 530 nM T35734 C91FRQ 44590935 IC50 > 2000 nM T35734 CM0L1S 44590936 IC50 = 49 nM T35734 CUV07Z 44590937 IC50 = 48 nM T35734 C79GTZ 44591877 IC50 = 128 nM T35734 CJ1H3Y 44591878 IC50 = 32 nM T35734 CA8B0N 44591879 IC50 = 37.2 nM T35734 CX5KL2 44591881 IC50 = 11 nM T35734 CP82ZQ 44591902 IC50 = 44.5 nM T35734 C1K3SI 44591911 IC50 = 49.1 nM T35734 C3UN7O 44591915 IC50 = 32.2 nM T35734 CH36JN 44591916 IC50 = 173 nM T35734 C9G7CU 44591917 IC50 = 28.7 nM T35734 CZP71X 44591919 IC50 = 200 nM T35734 CG9UZ0 44591920 IC50 = 33.6 nM T35734 C8STJ5 44591943 IC50 = 91.1 nM T35734 CMUT62 44591945 IC50 = 150 nM T35734 C1R8CA 44591947 IC50 = 164 nM T35734 CRN62E 44591948 IC50 = 52.1 nM T35734 CY1S6R 44591949 IC50 = 23.9 nM T35734 CRL8G0 44591950 IC50 = 200 nM T35734 COSI19 44591954 IC50 = 75.3 nM T35734 CXN28C 44591956 IC50 = 39.4 nM T35734 CDZ47K 44591957 IC50 = 35 nM T35734 CQ17WF 44591960 IC50 = 59.1 nM T35734 CGD1E7 44591962 IC50 = 54.1 nM T35734 CTUL67 44591963 IC50 = 12.7 nM T35734 C64ZKC 44593664 IC50 < 1 nM T35734 C01BFQ 44593665 IC50 = 3 nM T35734 CV3SC2 44626307 IC50 = 4 nM T35734 C54QWT 45267059 IC50 = 688 nM T35734 CUT2B4 45267348 IC50 = 333 nM T35734 C1O6IT 45267413 IC50 = 145 nM T35734 CJH3A2 45268206 IC50 = 5 nM T35734 C4WR0V 45269087 IC50 = 430 nM T35734 CRPS25 45269096 IC50 = 235 nM T35734 C7BNY6 45269104 IC50 = 7 nM T35734 C0RU3K 45269132 IC50 = 156 nM T35734 CS1Q2X 45269947 IC50 = 1100 nM T35734 C1BE5U 45269948 IC50 = 1100 nM T35734 CG1H9N 45269950 IC50 = 7.5 nM T35734 C6MI3J 45269972 IC50 = 240 nM T35734 CBHQ23 45269986 IC50 = 6.6 nM T35734 C2CQ1A 45270006 IC50 = 1.3 nM T35734 CI0XP7 45270738 IC50 = 1 nM T35734 C1NT2M 45270771 IC50 = 8400 nM T35734 CA05IG 45270778 IC50 = 11 nM T35734 CZ7MK9 45270788 IC50 = 10 nM T35734 C9TM2P 45271593 IC50 = 120 nM T35734 C06YAD 45271599 IC50 < 1 nM T35734 CG0I8P 45271610 IC50 = 187 nM T35734 C6FBH0 45271618 IC50 = 7 nM T35734 CEB59R 45272465 IC50 = 130 nM T35734 C71VIG 45272510 IC50 = 7 nM T35734 C05EDY 45272511 IC50 = 11 nM T35734 C5IB7N 45272559 IC50 = 42 nM T35734 CD62AH 45273373 IC50 = 480 nM T35734 CMN39U 45273380 IC50 = 14 nM T35734 CJVQ74 45366530 IC50 = 650 nM T35734 C08IRD 45426851 IC50 = 17 nM T35734 C8VR1Q 45484853 IC50 = 25 nM T35734 CO8R9W 45484854 IC50 = 1100 nM T35734 C5YV9X 45484856 IC50 = 8 nM T35734 C7UCG8 45484857 IC50 = 19 nM T35734 C0YUZ9 45484863 IC50 = 2500 nM T35734 CS0HE5 45484864 IC50 = 960 nM T35734 C38WJT 45484867 IC50 > 10000 nM T35734 C1MZ5G 45484868 IC50 = 19 nM T35734 CLG6I3 45484876 IC50 = 1200 nM T35734 CAZ38B 45484877 IC50 = 70 nM T35734 CKI5S0 45484887 IC50 > 10000 nM T35734 CEW57P 45484895 IC50 = 74 nM T35734 CI5P1N 45484901 IC50 = 470 nM T35734 C58XUK 45484924 IC50 > 10000 nM T35734 COJ60W 45484925 IC50 = 18 nM T35734 CF8XO4 45484926 IC50 = 91 nM T35734 C5GE7U 45484932 IC50 = 23 nM T35734 CTSI64 45484933 IC50 = 58 nM T35734 C9GBY0 45484940 IC50 = 4700 nM T35734 CDW0U7 45484941 IC50 > 10000 nM T35734 COKX69 45484942 IC50 = 40 nM T35734 CEMC68 45484943 IC50 = 8 nM T35734 C6WMO0 45484951 IC50 > 10000 nM T35734 C4GXF5 45484952 IC50 > 10000 nM T35734 CFO46G 45484953 IC50 = 27 nM T35734 CZK12H 45484954 IC50 = 31 nM T35734 CPD6F3 45484955 IC50 = 60 nM T35734 C5OJ2G 45484956 IC50 = 160 nM T35734 CSA13N 45484957 IC50 = 5200 nM T35734 CP9S8X 45484958 IC50 = 70 nM T35734 CSA5N3 45484959 IC50 = 4 nM T35734 CVB1L8 45484963 IC50 = 10 nM T35734 CZ4MY1 45484970 IC50 = 340 nM T35734 CMDA19 45487786 IC50 = 16 nM T35734 CKW7I6 45487791 IC50 = 21 nM T35734 C76IRB 45487797 IC50 = 5.4 nM T35734 C8UFN0 45487802 IC50 = 21 nM T35734 CJAP62 45487803 IC50 = 77 nM T35734 C93DRN 45487807 IC50 = 15 nM T35734 CK6VM4 45487814 IC50 = 66 nM T35734 C5WX4B 45487815 IC50 = 110 nM T35734 CSB52O 45487825 IC50 = 270 nM T35734 CR5W8V 45487826 IC50 = 31 nM T35734 C5ZYA0 45487831 IC50 = 4.6 nM T35734 CO2C7S 45487832 IC50 = 12 nM T35734 C79MYF 45487839 IC50 = 0.1 nM T35734 CBNV87 45487845 IC50 = 1500 nM T35734 C6RI7X 45487846 IC50 = 12 nM T35734 CG53MB 45724855 IC50 = 41 nM T35734 CBJ46X 45741848 IC50 = 6.9 nM T35734 CD3HM9 45754043 IC50 = 1200 nM T35734 CT5Q1F 45888834 IC50 = 0.4 nM T35734 CR7U6V 45889074 Ki = 0.49 nM T35734 CKQP51 46173998 Ki = 2000 nM T35734 C7F1LT 46224990 IC50 = 220 nM T35734 CTCH43 46225053 IC50 = 5.6 nM T35734 CR13CP 46225084 IC50 = 35 nM T35734 CEO34K 46225085 IC50 = 39 nM T35734 CZR0O7 46225086 IC50 = 17 nM T35734 C9WN8M 46225119 EC50 = 18 nM T35734 C2ZHI0 46225120 EC50 = 0.44 nM T35734 CW4DP1 46225121 EC50 = 0.63 nM T35734 C92EYK 46225159 EC50 = 0.78 nM T35734 C2K9HF 46225160 EC50 = 1.65 nM T35734 CHJE06 46225161 EC50 = 0.25 nM T35734 CB0J4D 46225162 EC50 = 0.97 nM T35734 CDBX78 46225163 EC50 = 0.34 nM T35734 CR23VF 46225206 EC50 = 0.29 nM T35734 C9JA2C 46700789 IC50 = 1 nM T35734 C43CHW 46743119 IC50 = 490 nM T35734 C5I8ML 46871778 IC50 = 4 nM T35734 C2LMI8 46871779 IC50 = 14 nM T35734 CRU1P2 46882874 IC50 = 7 nM T35734 CYU8X6 46882875 IC50 = 7 nM T35734 CX5CZ7 46882876 IC50 = 29 nM T35734 C0FM2D 46882917 IC50 < 1000 nM T35734 CC1VO9 46882918 IC50 = 52 nM T35734 C27RIV 46882919 IC50 = 5 nM T35734 CE3O7D 46882949 IC50 < 1000 nM T35734 CHS1X0 46882950 IC50 = 1.3 nM T35734 C3S9WE 46882951 IC50 = 5 nM T35734 C3A1ZF 46882969 IC50 = 12 nM T35734 CG3D0K 46882971 IC50 = 1.4 nM T35734 CD7XA2 46882972 IC50 = 5 nM T35734 CY5CW2 46882973 IC50 = 3 nM T35734 C3ZPY7 46882986 IC50 < 1000 nM T35734 CKX8N2 46882987 IC50 < 1000 nM T35734 CG81CZ 46882988 IC50 = 12 nM T35734 CP87CA 46883032 IC50 < 1000 nM T35734 CWU4T2 46883033 IC50 = 30 nM T35734 C41RYD 46883034 IC50 = 28 nM T35734 C3SQ2Z 46883035 IC50 = 19 nM T35734 CS51UC 46883473 IC50 = 550 nM T35734 CL0S4B 46883474 IC50 = 7 nM T35734 C0K5ZJ 46883508 IC50 = 8 nM T35734 CMNJ24 46883509 IC50 = 14 nM T35734 CF4VC1 46883510 IC50 < 1000 nM T35734 CTCH12 46888804 IC50 = 68 nM T35734 C82VNT 46888805 IC50 = 280 nM T35734 C51WUS 46888844 IC50 = 62 nM T35734 CCY7L2 46888845 IC50 = 2800 nM T35734 CT62BY 46888846 IC50 = 130 nM T35734 C1O6HF 46888847 IC50 = 22 nM T35734 C2VG0D 46888848 IC50 = 18 nM T35734 C2XAN5 46888872 IC50 = 110 nM T35734 CD7P3L 46888913 IC50 = 760 nM T35734 CB9VZ6 46888914 IC50 = 38 nM T35734 CH1N7A 46888915 IC50 = 18 nM T35734 CTX25Y 46888916 IC50 = 490 nM T35734 CYFL60 46888977 IC50 = 19 nM T35734 C6HA8X 46888978 IC50 = 80 nM T35734 C4Z5AO 46888979 IC50 = 20 nM T35734 C39LBN 46889036 IC50 = 48 nM T35734 C1V7OZ 46889037 IC50 = 19 nM T35734 CPM6B0 46889038 IC50 = 3 nM T35734 CZ5AQ1 46889055 IC50 = 140 nM T35734 CD1TG4 46889056 IC50 = 16 nM T35734 CPLF71 46889057 IC50 = 1 nM T35734 CL08OY 46889083 IC50 = 8 nM T35734 CU62DM 46889110 IC50 = 3 nM T35734 CHW72U 46889111 IC50 = 54 nM T35734 C5J4XI 46889138 IC50 = 19 nM T35734 C1ZTX8 46889139 IC50 = 12 nM T35734 C8WE0H 46889165 IC50 = 54 nM T35734 CUG5H3 46889204 IC50 = 1 nM T35734 C3YMK6 46889226 IC50 = 1 nM T35734 CM35UH 46889249 IC50 = 800 nM T35734 C9JP2D 46889270 IC50 = 120 nM T35734 C1DW4T 46889271 IC50 = 130 nM T35734 C73MTG 46889272 IC50 = 27 nM T35734 C7QIT8 46891216 IC50 = 3 nM T35734 CW7R5O 46891217 IC50 = 7 nM T35734 CSIX69 46891218 IC50 = 9 nM T35734 C7YTV8 46933844 IC50 = 9100 nM T35734 C9FUJ7 47039916 IC50 = 12.3 nM T35734 CUXM58 47103132 IC50 = 116 nM T35734 C4EJ8R 47103446 IC50 = 386.1 nM T35734 CP74XN 47103624 IC50 = 485 nM T35734 CY34GV 47171960 IC50 = 16.6 nM T35734 CZLG95 47193806 IC50 = 56.2 nM T35734 CO6VB1 47760732 IC50 = 1551 nM T35734 CMVH81 49120644 IC50 = 6.7 nM T35734 C8TLK6 49780161 IC50 = 0.4 nM T35734 C2KWR9 49780162 IC50 = 17 nM T35734 CT0RZ7 49780165 IC50 = 0.6 nM T35734 CU71PT 49780166 IC50 = 1.5 nM T35734 C0VP9D 49780366 IC50 = 0.5 nM T35734 C6E7IY 49780367 IC50 = 0.4 nM T35734 C0RI6X 49780368 IC50 = 0.5 nM T35734 C6K9PQ 49780369 IC50 = 0.4 nM T35734 CH2W5P 49780370 IC50 = 1.8 nM T35734 C5NP0F 49780576 IC50 = 0.4 nM T35734 C0Q8IU 49780577 IC50 = 0.8 nM T35734 CO0WZ3 49782571 IC50 = 2.7 nM T35734 CS3CD2 49782795 IC50 = 3 nM T35734 CR59XD 49782796 IC50 = 3800 nM T35734 CJWD97 49782800 IC50 = 8.3 nM T35734 CC6I9P 49782801 IC50 = 2.8 nM T35734 C61CTM 49782802 IC50 = 87 nM T35734 CV7LP3 49783004 IC50 = 3.5 nM T35734 C6CPO0 49783005 IC50 = 61 nM T35734 CSR30T 49783006 IC50 > 5000 nM T35734 C9PA2V 49783007 IC50 = 2000 nM T35734 C84NCM 49783008 IC50 = 38 nM T35734 CMK46W 49783009 IC50 = 140 nM T35734 CC6WS5 49783010 IC50 = 330 nM T35734 CDVQ35 49783213 IC50 = 406 nM T35734 CD32IR 49783214 IC50 = 79 nM T35734 CS26JG 49783215 IC50 = 10 nM T35734 C2I1XR 49783216 IC50 = 3.6 nM T35734 CXR8H0 49783217 IC50 = 7.2 nM T35734 CD3FU8 49783218 IC50 = 39 nM T35734 CTX12F 49783219 IC50 = 300 nM T35734 CH4A8W 49783220 IC50 = 21 nM T35734 CO9PT0 49783422 IC50 = 1100 nM T35734 C7BWD6 49783423 IC50 = 3.4 nM T35734 C7G9JE 49783424 IC50 = 0.4 nM T35734 C3C9US 49783425 IC50 > 5000 nM T35734 CYS9I4 49783426 IC50 = 4.1 nM T35734 C1KAG5 49783427 IC50 = 0.7 nM T35734 C0GU3S 49783428 IC50 = 17 nM T35734 C90AKU 49837852 IC50 = 562.34 nM T35734 CAU59E 49837853 IC50 = 6.1 nM T35734 C3QXR1 49850586 IC50 = 21.5 nM T35734 C8S6UB 49850587 IC50 = 91.4 nM T35734 CXE5N8 49850686 IC50 = 5.4 nM T35734 CLN9O1 49850687 IC50 = 1.8 nM T35734 C45FVD 49850688 IC50 = 1.4 nM T35734 CYHB45 49850689 IC50 = 1 nM T35734 CT1R3P 49850690 IC50 = 9.6 nM T35734 CE1XO5 49850788 IC50 = 13.6 nM T35734 CZ95TG 49850789 IC50 = 3.3 nM T35734 CCY01S 49850890 IC50 = 7.8 nM T35734 CAIY43 49850891 IC50 = 2880 nM T35734 C2RY8O 49850892 IC50 = 23.1 nM T35734 C4GJ3F 49850893 IC50 = 17.9 nM T35734 C6BN9J 49850894 IC50 = 5290 nM T35734 C1P0RQ 49851001 IC50 = 13.3 nM T35734 CI54KF 49851002 IC50 = 44.8 nM T35734 C8RGD1 49851003 IC50 = 11.5 nM T35734 C6MK7A 49851004 IC50 = 2.8 nM T35734 CX7G4B 49851005 IC50 = 39.4 nM T35734 CI8L1C 49851095 IC50 = 2.9 nM T35734 CQ5X1H 49851096 IC50 = 14.6 nM T35734 CG9L4Z 49851097 IC50 = 16.5 nM T35734 CRZ97Q 49851098 IC50 = 7.1 nM T35734 CVY8Z1 49851099 IC50 = 20.1 nM T35734 C2ZDI0 49851178 IC50 = 11.7 nM T35734 CH41EK 49851179 IC50 = 67.1 nM T35734 C5F3DW 49851180 IC50 = 97460 nM T35734 CJ3Y8D 49851181 IC50 = 27.2 nM T35734 C8TVC6 49851182 IC50 = 156 nM T35734 C8LP4Q 49851275 IC50 = 72770 nM T35734 C41ZNW 49851276 IC50 = 14.8 nM T35734 C8C2OF 49851277 IC50 = 126 nM T35734 C27MRX 49851278 IC50 = 13.8 nM T35734 COZ96T 49851279 IC50 = 6 nM T35734 CKE92W 49851383 IC50 = 994 nM T35734 CI6UW1 49851384 IC50 = 3.6 nM T35734 C09EFL 49851385 IC50 = 3.3 nM T35734 C0DR3Y 49851386 IC50 = 3150 nM T35734 C6N4YQ 49851387 IC50 = 2.7 nM T35734 CY9B6U 49851483 IC50 = 7 nM T35734 CMU9I0 49851484 IC50 = 2.8 nM T35734 C8LA9S 50899467 IC50 = 4.7 nM T35734 CO64EX 50899554 IC50 = 8.8 nM T35734 CW3T2O 50916358 IC50 = 45 nM T35734 C1GEQ8 50916359 IC50 = 199 nM T35734 CIN13F 50916540 IC50 = 192 nM T35734 CZEC61 50916541 IC50 = 230 nM T35734 CG8E0B 50916542 IC50 = 185 nM T35734 C1XLQ4 50916543 IC50 = 108 nM T35734 CGL49J 50916713 IC50 = 26 nM T35734 C10VRU 50916714 IC50 = 16 nM T35734 CJ19FC 50916715 IC50 = 6.7 nM T35734 C5K6SO 50916716 IC50 = 42 nM T35734 CE96RK 50916901 IC50 = 130 nM T35734 C0V1UC 50916902 IC50 = 186 nM T35734 C8ZH9S 50916903 IC50 = 3 nM T35734 CF3H2U 50916904 IC50 = 58 nM T35734 C4C6TQ 50917098 IC50 = 23 nM T35734 CH96SZ 50917101 IC50 = 24 nM T35734 CFIA61 50917102 IC50 = 3.4 nM T35734 CD6XP3 50917281 IC50 = 1.9 nM T35734 C3MZ8U 50917282 IC50 = 41 nM T35734 CF3N1Z 50917284 IC50 = 21 nM T35734 CXBU71 50917285 IC50 = 46 nM T35734 CN50GR 50917629 IC50 = 0.96 nM T35734 CEP59A 51050039 IC50 = 61.66 nM T35734 COB7S2 51050040 IC50 = 39.81 nM T35734 C4RK2I 51050041 IC50 = 30.2 nM T35734 CVE5Y2 51050042 IC50 = 2.291 nM T35734 CQW72U 51188664 IC50 = 1.2 nM T35734 C75KEO 52546186 IC50 = 13 nM T35734 C1SO7D 52546187 IC50 = 13 nM T35734 CTL4U3 52641320 IC50 = 1510 nM T35734 CT50NH 52641321 IC50 = 332 nM T35734 CA8N9P 52911994 IC50 = 22 nM T35734 CY6EO0 52940693 IC50 = 21 nM T35734 CTS9H0 52942123 IC50 = 1 nM T35734 CR40WN 52944428 IC50 = 7.3 nM T35734 CF58QT 52946747 IC50 = 28 nM T35734 CKLW43 52948184 IC50 = 650 nM T35734 CNM5Y9 52949345 IC50 = 23 nM T35734 C6DF9H 52951272 IC50 = 88 nM T35734 C6VWE2 52951275 IC50 = 26 nM T35734 CD8SA7 52951485 IC50 = 25 nM T35734 CH1T5N 52951486 IC50 = 2.6 nM T35734 CPU67E 52951487 IC50 = 47 nM T35734 CBN86G 52951488 IC50 = 6 nM T35734 CYZ4C6 52951489 IC50 = 110 nM T35734 C51QFH 52951612 IC50 = 72 nM T35734 CRH4E8 52951613 IC50 = 84 nM T35734 CPTE73 52951614 IC50 = 32 nM T35734 C9HUZ2 52951734 IC50 = 3.4 nM T35734 C96TVC 52951735 IC50 = 4.1 nM T35734 CLN12R 52951736 IC50 = 10 nM T35734 C7GFM3 52951862 IC50 = 1550 nM T35734 CFJQ74 52951863 IC50 = 0.8 nM T35734 CUSD82 52951864 IC50 = 0.5 nM T35734 CP6M1R 52951865 IC50 = 0.5 nM T35734 CD32FZ 52951866 IC50 = 0.8 nM T35734 CU51RA 52951990 IC50 = 0.9 nM T35734 CDT5Z6 52951991 IC50 = 0.5 nM T35734 CD46ZG 53317560 IC50 = 4.677 nM T35734 CJD3W2 53317889 IC50 = 25 nM T35734 C7LIV0 53317890 IC50 = 6 nM T35734 CUS63Y 53320344 IC50 = 270 nM T35734 CP7Z2K 53321845 IC50 = 120 nM T35734 C79LEC 53323157 IC50 = 58 nM T35734 CZ7U6E 53323158 IC50 = 14 nM T35734 C6UBQ1 54672302 IC50 = 8600 nM T35734 CQ9W1N 54672377 IC50 = 5200 nM T35734 CP1M5C 54752297 IC50 = 0.4 nM T35734 C43YCF 54878877 IC50 > 10000 nM T35734 CQ98UD 56054771 IC50 = 263 nM T35734 CN41ZQ 56659144 IC50 = 12 nM T35734 CVLG75 56662646 IC50 = 1.6 nM T35734 C6HOT7 56664970 IC50 = 0.4 nM T35734 C20MUR 56666108 IC50 = 1 nM T35734 C2O8FJ 56666109 IC50 = 0.4 nM T35734 C47YSD 56666110 IC50 = 1838.1 nM T35734 CFM0U7 56666111 IC50 = 260.4 nM T35734 CIRX84 56669513 IC50 = 14.8 nM T35734 CI5GV0 56669514 IC50 = 6.4 nM T35734 C5TKW3 56669515 IC50 = 0.5 nM T35734 CQX08R 56669516 IC50 = 0.4 nM T35734 CJ1XC6 56669517 IC50 = 3.7 nM T35734 C5TXU2 56669518 IC50 = 38.1 nM T35734 CEVF80 56669519 IC50 = 524.8 nM T35734 C7A6BI 56669520 IC50 = 242.6 nM T35734 C25SEN 56673015 IC50 = 1.1 nM T35734 CG2D0W 56673016 IC50 = 24.2 nM T35734 CRY08V 56673017 IC50 = 463.8 nM T35734 CBI9X3 56676336 IC50 = 0.4 nM T35734 C8QZ2J 56676337 IC50 = 0.4 nM T35734 CBK8Q7 56676338 IC50 = 4.5 nM T35734 CN0KH6 56676339 IC50 = 1.9 nM T35734 CV90OL 56676340 IC50 = 4.8 nM T35734 C7HKP9 56679661 IC50 = 0.4 nM T35734 C57YQT 56679662 IC50 = 0.4 nM T35734 C5OX8U 56682986 IC50 = 0.4 nM T35734 CV4MY1 56682987 IC50 = 0.4 nM T35734 CG1N9O 56838295 IC50 = 59 nM T35734 CT2KM8 56968119 Ki = 0.98 nM T35734 CE2MO3 56968120 Ki = 1.22 nM T35734 CK3EI1 56968121 Ki = 1.79 nM T35734 CX8P2K 56971637 Ki = 0.43 nM T35734 CN3C5U 56971638 Ki = 2.23 nM T35734 CM98ZO 56971639 Ki = 0.37 nM T35734 CC94ZX 56971640 Ki = 1.2 nM T35734 CT58YR 56971641 Ki = 1.74 nM T35734 C08KOV 56971642 Ki = 1.47 nM T35734 C5Z2IQ 57391544 IC50 = 7.7 nM T35734 CA4M3J 57391545 IC50 = 56 nM T35734 CGAN95 57391578 IC50 = 16 nM T35734 CWS0V6 57391579 IC50 = 4200 nM T35734 CUE29O 57391580 IC50 = 1200 nM T35734 CZMR95 57391641 IC50 = 22 nM T35734 C6VH9T 57391642 IC50 = 960 nM T35734 CWP8B0 57391643 IC50 = 450 nM T35734 C7PED9 57391644 IC50 = 1300 nM T35734 CTQM58 57393386 IC50 = 490 nM T35734 CL39PS 57393387 IC50 = 12 nM T35734 C3IO1Y 57393388 IC50 = 1100 nM T35734 C4H3NU 57395026 IC50 = 12 nM T35734 C2KXA3 57395056 IC50 = 2000 nM T35734 CG7MX1 57395107 IC50 = 950 nM T35734 CL9YH2 57395108 IC50 = 24 nM T35734 CORG37 57395109 IC50 = 2100 nM T35734 C8Q9PF 57396875 IC50 = 46.1 nM T35734 CNY05K 57396876 IC50 = 6.7 nM T35734 C9UVW6 57396877 IC50 = 150 nM T35734 CT9Y6C 57396878 IC50 = 50000 nM T35734 CLZ96T 57398545 IC50 = 27 nM T35734 CKU24F 57398580 IC50 = 17 nM T35734 C5EF6K 57398581 IC50 = 6000 nM T35734 CV94HG 57398635 IC50 = 120 nM T35734 CDW1L7 57400244 IC50 = 120 nM T35734 C5TG7I 57400245 IC50 = 35 nM T35734 CQ0N8R 57400246 IC50 = 630 nM T35734 C4PG6X 57400247 IC50 = 780 nM T35734 CB93CS 57400302 IC50 = 340 nM T35734 C1GO8X 57400303 IC50 = 240 nM T35734 C59RZQ 57400304 IC50 = 5.4 nM T35734 CSE09D 57400305 IC50 = 18 nM T35734 C0OUD9 57402048 IC50 = 1700 nM T35734 C8KTV0 57402049 IC50 = 150 nM T35734 C62UPT 57402050 IC50 = 2000 nM T35734 CVU92Z 57402112 IC50 = 13000 nM T35734 C41UIG 57403792 IC50 = 6000 nM T35734 CN01AK 57403793 IC50 = 9.6 nM T35734 C6UK4X 57403794 IC50 = 21 nM T35734 CEH4X2 57403858 IC50 = 140 nM T35734 CE70AJ 57403859 IC50 = 15 nM T35734 CX4CP8 57551019 IC50 = 7 nM T35734 C0P8SB 58758181 IC50 = 74.2 nM T35734 C8TQ4C 59168587 IC50 = 6.3 nM T35734 CMTY65 59168602 IC50 = 67 nM T35734 C70QYO 59168631 IC50 = 1.8 nM T35734 CI1U7Q 59168635 IC50 = 3 nM T35734 CLK40I 59168639 IC50 = 2.7 nM T35734 CQ4YH6 59168644 IC50 = 1.3 nM T35734 C0YIP3 59168645 IC50 = 10.8 nM T35734 CB2T5D 59168647 IC50 = 4 nM T35734 CY0HA2 59168653 IC50 = 4.1 nM T35734 CZ0S2A 59168654 IC50 = 2.3 nM T35734 C2JYD4 59168656 IC50 = 3.8 nM T35734 CS24XA 59168659 IC50 = 1.6 nM T35734 CPQ4S8 59168665 IC50 = 1 nM T35734 CI81KY 59168676 IC50 = 0.9 nM T35734 CJKW13 59168698 IC50 = 0.6 nM T35734 C19EIV 59168699 IC50 = 12 nM T35734 CAXR35 59168701 IC50 = 0.8 nM T35734 C0B2WK 59168704 IC50 = 2.4 nM T35734 CMA9G5 59168740 IC50 = 1.2 nM T35734 CC4Y0T 59168741 IC50 = 1.6 nM T35734 CLCK72 59168751 IC50 = 12.1 nM T35734 CMG7L3 59168758 IC50 = 5.1 nM T35734 CN1US8 59447733 IC50 = 3 nM T35734 C9S4DU 59447737 IC50 = 4 nM T35734 C2O9UC 59595168 IC50 = 400 nM T35734 C2JCP7 59688918 IC50 = 5.2 nM T35734 CU67VY 60022915 IC50 = 67 nM T35734 C9W0PE 60150671 IC50 = 0.5 nM T35734 C7ML8X 60162803 IC50 = 6.8 nM T35734 C6HTG5 60162804 IC50 = 142 nM T35734 COR6K2 60162931 IC50 = 7.3 nM T35734 CV2DK1 60162932 IC50 = 133.4 nM T35734 C06RYB 60162933 IC50 = 46.3 nM T35734 CZ0DQ8 60163072 IC50 = 41.8 nM T35734 C4X2BC 60163073 IC50 = 0.5 nM T35734 CT9LE2 60163074 IC50 = 9 nM T35734 C47NMI 60163075 IC50 = 1 nM T35734 C34XUR 60165328 IC50 = 63 nM T35734 CW3G6N 60196633 IC50 = 0.5 nM T35734 CUV14K 60196634 IC50 = 0.5 nM T35734 CU32ED 60196737 IC50 = 0.5 nM T35734 CKB59I 60196738 IC50 = 0.5 nM T35734 C40LVZ 60196740 IC50 = 0.5 nM T35734 CMPK13 60196846 IC50 = 5 nM T35734 C5EUK3 60638849 IC50 = 0.5 nM T35734 CJ6KY4 66556109 IC50 > 500 nM T35734 CN1YJ7 66556282 IC50 = 255 nM T35734 CNR87G 66556283 IC50 > 500 nM T35734 CQ8NR5 66556284 IC50 > 500 nM T35734 CUF17E 66556285 IC50 > 500 nM T35734 CU81GD 66556287 IC50 = 71 nM T35734 C9ZN0A 66556446 IC50 > 500 nM T35734 CS29OQ 66556448 IC50 = 57 nM T35734 C5QUB6 66556450 IC50 = 96 nM T35734 CW0BJ8 66556451 IC50 = 32 nM T35734 CJ62RI 66556452 IC50 = 22 nM T35734 CXD3F5 66556453 IC50 = 11 nM T35734 C3W8EJ 66556614 IC50 = 6 nM T35734 COG08Y 66556615 IC50 = 32 nM T35734 C37SQB 66556616 IC50 = 23 nM T35734 CCU1N2 66556617 IC50 > 500 nM T35734 CFW4B3 66556618 IC50 = 11 nM T35734 CC64RF 66556619 IC50 > 500 nM T35734 CP0Z1F 66556620 IC50 = 32 nM T35734 CS27JO 66556784 IC50 = 57 nM T35734 C91SQJ 66556786 IC50 = 10 nM T35734 CH6I2G 66556787 IC50 > 500 nM T35734 CX76QT 66556789 IC50 = 41 nM T35734 C8ON5H 66556969 IC50 = 282 nM T35734 CBZL92 66556970 IC50 > 500 nM T35734 CB6YQ9 66556971 IC50 > 500 nM T35734 CI8HN5 66556972 IC50 > 500 nM T35734 CW17YX 68281294 IC50 = 0.5 nM T35734 CAZM23 68329420 IC50 = 650 nM T35734 C0A6TK 70681638 IC50 = 1.7 nM T35734 CCH7S4 70682540 IC50 = 1160 nM T35734 CDT78V 70683764 IC50 = 1.5 nM T35734 C5TP4N 70683777 IC50 = 4.7 nM T35734 C9HL5Y 70685919 IC50 = 3.8 nM T35734 CL8YK9 70688033 IC50 = 25.8 nM T35734 C40EKD 70688854 IC50 = 9 nM T35734 CYO5N2 70689719 EC50 = 1.7 nM T35734 CEJ64G 70690062 IC50 = 13.6 nM T35734 C42DPF 70690068 IC50 = 3.3 nM T35734 C7OG0W 70690074 IC50 = 6.1 nM T35734 CI58YH 70692220 IC50 = 8.2 nM T35734 CYG96X 70693911 EC50 = 23 nM T35734 CO7NS3 70694280 IC50 = 3.1 nM T35734 C64RNI 70694281 IC50 = 2.6 nM T35734 C47OKG 70694285 IC50 = 66.5 nM T35734 CG2M1A 70694286 IC50 = 6.2 nM T35734 CSEP-96 70696372 IC50 = 1.6 nM T35734 CRQ5K6 71450212 IC50 = 252 nM T35734 CK6C4E 71452039 IC50 = 747 nM T35734 C2P3VJ 71453182 IC50 = 25000 nM T35734 CR23KT 71453845 IC50 = 39 nM T35734 C3I8ZX 71453846 IC50 = 2009 nM T35734 C0YQW3 71455576 IC50 = 1923 nM T35734 C7D9PO 71457365 IC50 = 23 nM T35734 C8D5FS 71457366 IC50 = 43 nM T35734 CLO6U1 71457367 IC50 = 46 nM T35734 CH25YT 71457368 IC50 = 611 nM T35734 C98QRS 71457369 IC50 = 178 nM T35734 CY3J1I 71457370 IC50 = 73 nM T35734 CK9YX1 71457371 IC50 = 258 nM T35734 CPQ72D 71459225 IC50 = 27 nM T35734 C9M1XP 71459226 IC50 = 87 nM T35734 CW7NR3 71459227 IC50 = 304 nM T35734 CGF67V 71462737 IC50 = 943 nM T35734 C2GMD4 71487912 IC50 = 1600 nM T35734 C5X4QS 71522732 IC50 = 0.4 nM T35734 CJP36F 71540714 IC50 = 0.4 nM T35734 CQKY73 71540830 IC50 = 25 nM T35734 CGO4I7 71540946 IC50 = 55 nM T35734 CG30QP 71540947 IC50 = 13 nM T35734 C9RBG2 71540948 IC50 = 110 nM T35734 C13GIH 71541063 IC50 = 29 nM T35734 CL47IS 71541161 IC50 = 20 nM T35734 C4FGD8 71541162 IC50 = 43 nM T35734 CJ89SB 71541261 IC50 = 1.6 nM T35734 CL0T4N 71541262 IC50 = 78 nM T35734 C2BI5Q 71541378 IC50 = 0.6 nM T35734 COBG71 71541379 IC50 = 30000 nM T35734 COP06B 71566536 IC50 = 0.3 nM T35734 C2SA5M 71566537 IC50 = 0.4 nM T35734 C1XF4C 71566538 IC50 = 0.3 nM T35734 CCZ3A4 71574951 IC50 = 106 nM T35734 CT7I1M 71574952 IC50 = 65 nM T35734 CR45LK 71575134 IC50 = 70 nM T35734 C9L4OE 71575135 IC50 = 44 nM T35734 C1J8ZR 71575136 IC50 = 32 nM T35734 C6XA4W 71575233 IC50 = 30 nM T35734 C8A5YG 71575234 IC50 = 82 nM T35734 C6XR5B 71575235 IC50 = 52 nM T35734 C47GVA 71575236 IC50 = 71 nM T35734 CK0W3S 71575346 IC50 = 70 nM T35734 CIK2H4 71575347 IC50 = 147 nM T35734 CPX09S 71575348 IC50 = 201 nM T35734 C6O7LP 71575349 IC50 = 92 nM T35734 C5CLE8 71575350 IC50 = 42 nM T35734 CC0D1M 71575458 IC50 = 104 nM T35734 CE0TN5 71575459 IC50 = 38 nM T35734 C1XA7Z 71575460 IC50 = 38 nM T35734 C61AXK 71575461 IC50 = 62 nM T35734 C5C3SP 71575560 IC50 = 189 nM T35734 CI7K0M 71575561 IC50 = 100 nM T35734 CQU1T8 71575562 IC50 = 242 nM T35734 CEG4J2 71579507 IC50 = 2670 nM T35734 CWF10M 71579508 IC50 = 3020 nM T35734 CQ16DL 71579510 IC50 = 1720 nM T35734 CPOI89 71579596 IC50 = 3000 nM T35734 C7FLP0 71579600 IC50 = 1070 nM T35734 CFK0L9 71580977 IC50 = 17200 nM T35734 C2TDO9 71580978 IC50 = 16400 nM T35734 CH9RI8 71602741 IC50 = 19 nM T35734 C0XB6Y 71602742 IC50 = 7 nM T35734 CY65GE 71602743 IC50 = 292 nM T35734 CVS2D6 71602744 IC50 = 13 nM T35734 CSM9Q0 71602794 IC50 = 31 nM T35734 C5AG1N 71602842 IC50 = 24010 nM T35734 CP93VJ 71602843 IC50 = 775 nM T35734 COW9S6 71602844 IC50 = 79 nM T35734 CAYQ70 71602845 IC50 = 1012 nM T35734 C5RN6H 71602846 IC50 = 948 nM T35734 CKQ83N 71602847 IC50 = 46 nM T35734 CDE61N 71602889 IC50 = 56 nM T35734 CB03OJ 71602890 IC50 = 0.8 nM T35734 CJZM10 71602891 IC50 = 117 nM T35734 C2BYG3 71602892 IC50 = 2 nM T35734 CU74KG 71602893 IC50 = 0.5 nM T35734 C74JHR 71602894 IC50 = 25 nM T35734 CP3G4L 71602941 IC50 = 20 nM T35734 CNT50S 71602942 IC50 = 595 nM T35734 CU10HM 71602943 IC50 = 557 nM T35734 CG5D7F 71602993 IC50 = 503 nM T35734 CWUG96 71602994 IC50 = 241 nM T35734 C3Q1UK 71602995 IC50 = 1575 nM T35734 CJ82BV 71602996 IC50 = 884 nM T35734 CXD8P9 71602997 IC50 = 2512 nM T35734 C6NP0U 71602998 IC50 = 751 nM T35734 C90GEU 71602999 IC50 = 488 nM T35734 CWV0L3 71603055 IC50 = 46 nM T35734 CENG10 71603056 IC50 = 73 nM T35734 CU6W9M 71603057 IC50 = 5 nM T35734 C0O7LX 71603058 IC50 = 710 nM T35734 C4G6RH 71603059 IC50 = 843 nM T35734 C0XCL7 71603060 IC50 = 2408 nM T35734 C36AGK 71603061 IC50 = 382 nM T35734 C2B5ZM 71603118 IC50 = 2463 nM T35734 C5VF1X 71603119 IC50 = 936 nM T35734 CCUW57 71655311 IC50 = 126 nM T35734 CN13KW 71655312 IC50 = 1585 nM T35734 CHR1L4 71655313 IC50 = 100 nM T35734 CHZ0U6 71655314 IC50 = 32 nM T35734 CXT60O 71655374 IC50 = 1 nM T35734 C9AIJ7 71655375 IC50 = 200 nM T35734 CGLA96 71655376 IC50 = 1600 nM T35734 C8OX4Q 71655377 IC50 = 630 nM T35734 C49YGB 71655378 IC50 = 400 nM T35734 CH7KA2 71655379 IC50 = 200 nM T35734 C39HIB 71655380 IC50 = 80 nM T35734 CG9P3O 71655442 IC50 = 1 nM T35734 CXW48Z 71655443 IC50 = 16 nM T35734 CM2P0R 71655444 IC50 = 1 nM T35734 CSP95X 71655445 IC50 = 1 nM T35734 C2PL3H 71655503 IC50 = 1 nM T35734 CWT6O7 71657834 IC50 = 392 nM T35734 C3VIY5 71660815 IC50 = 1.1 nM T35734 CN80BS 71678005 Ki = 0.31 nM T35734 C7GP1H 71678006 Ki = 1.23 nM T35734 CSK5G3 71678007 Ki = 0.99 nM T35734 C8JO9C 71678008 Ki = 1.17 nM T35734 C83QIH 71678169 Ki = 2.44 nM T35734 CE4TK5 71679326 Ki = 0.44 nM T35734 C08BPE 71679327 Ki = 0.19 nM T35734 CSG98X 71679344 IC50 = 1.4 nM T35734 CL68DC 71679345 IC50 = 1.9 nM T35734 C7A3GW 71679346 IC50 = 0.6 nM T35734 CM56VG 71679347 IC50 = 0.7 nM T35734 C89BYZ 71679348 IC50 = 0.125 nM T35734 C5W3AK 71679516 IC50 = 0.6 nM T35734 C2O6SX 71679518 IC50 = 0.5 nM T35734 C3JRL9 71679671 IC50 = 1.1 nM T35734 CE1V6I 71679838 IC50 = 0.4 nM T35734 C1NJQ5 71680197 Ki = 0.36 nM T35734 CC8M7Z 71680510 Ki = 0.22 nM T35734 CT93OP 71682347 IC50 = 0.5 nM T35734 C3NV9Q 71682348 IC50 = 8.6 nM T35734 CN7M9G 71682349 IC50 = 1 nM T35734 C8KU4O 71682499 IC50 = 0.5 nM T35734 C0XEQ1 71682500 IC50 = 0.5 nM T35734 CH81LG 71719756 IC50 = 6900 nM T35734 CP3RQ0 71730150 IC50 = 2 nM T35734 C8OT1D 72195347 IC50 = 0.4 nM T35734 CD1OS5 72374646 IC50 = 3 nM T35734 C6KVI9 72374647 IC50 = 0.7 nM T35734 C40LUJ 72374648 IC50 = 1.2 nM T35734 CFZX16 72374649 IC50 = 0.3 nM T35734 CA8KR5 72374650 IC50 = 0.5 nM T35734 CEVJ40 72374651 IC50 = 1.3 nM T35734 CSO1H8 72374760 IC50 = 0.6 nM T35734 C90VDO 72374761 IC50 = 0.6 nM T35734 C65BSO 72374762 IC50 = 0.8 nM T35734 C6K4RO 72374763 IC50 = 0.4 nM T35734 CK1M6B 72375936 IC50 = 175.6 nM T35734 C6R9AU 72375937 IC50 > 200 nM T35734 CE25VH 72375938 IC50 = 466.3 nM T35734 CKN49R 72375939 IC50 = 151.6 nM T35734 CJYH75 72375940 IC50 = 51.7 nM T35734 CO34RZ 72376037 IC50 = 6.7 nM T35734 C4Z7UC 72376038 IC50 = 5.7 nM T35734 CT5P8I 72376039 IC50 = 16.1 nM T35734 CIP34N 72376040 IC50 = 35.3 nM T35734 C32VEW 72376041 IC50 = 1.1 nM T35734 C60HTM 72376042 IC50 = 3.5 nM T35734 CS24KN 72376130 IC50 = 3.4 nM T35734 CQ4B1Z 72376131 IC50 = 115 nM T35734 C4QIT9 72376132 IC50 = 0.7 nM T35734 CJ4R7D 72376133 IC50 = 0.2 nM T35734 C8N5ZP 72376134 IC50 = 0.3 nM T35734 C8ERC3 72376135 IC50 = 0.2 nM T35734 C5M4KO 72376211 IC50 = 0.8 nM T35734 C39JDL 72376212 IC50 = 0.4 nM T35734 C7TD6E 72376213 IC50 = 0.2 nM T35734 CNY83E 72376214 IC50 = 0.5 nM T35734 C5YLR4 72376215 IC50 = 0.9 nM T35734 CP9BN5 72376216 IC50 = 2.8 nM T35734 CDKL42 73212758 IC50 = 5.4 nM T35734 CZW68P 73212763 IC50 = 2.96 nM T35734 C45PLS 73212854 IC50 = 1.3 nM T35734 C67FXY 73212855 IC50 = 3.2 nM T35734 CQ75VH 73212856 IC50 = 1.4 nM T35734 CBVL82 73212857 IC50 = 1.2 nM T35734 C2KMT6 73212858 IC50 = 1 nM T35734 C3DJ7O 73212859 IC50 = 0.8 nM T35734 CL4H3S 73212938 IC50 = 5.4 nM T35734 CN39QV 73212939 IC50 = 4.2 nM T35734 CQ1EH0 73212940 IC50 = 0.9 nM T35734 CE3U5B 73212941 IC50 = 1.8 nM T35734 CM3Y1O 73212942 IC50 = 2.9 nM T35734 CT3FE1 73212943 IC50 = 2.1 nM T35734 CDJ9S2 73213026 IC50 = 0.6 nM T35734 C0RB2F 73213027 IC50 = 0.7 nM T35734 CN14LK 73346169 IC50 = 220 nM T35734 CX3WF4 73346170 IC50 = 22256 nM T35734 CIB20T 73347696 IC50 = 13607 nM T35734 C8RN3I 73349215 IC50 = 275 nM T35734 C6G5RM 73349216 IC50 = 16699 nM T35734 CG4RW9 73350796 IC50 = 269 nM T35734 CQOD98 73353501 IC50 = 0.7 nM T35734 CQTW58 73353751 IC50 = 224 nM T35734 CA48NE 73355280 IC50 = 3471 nM T35734 C1NUB8 73355283 IC50 = 10082 nM T35734 CT97QR 73669466 IC50 = 50 nM T35734 CK87OC 73669627 IC50 = 4.4 nM T35734 C8FN6P 73669628 IC50 = 1.2 nM T35734 CRKE04 76310125 IC50 > 10000 nM T35734 C4NH2U 76310126 IC50 > 10000 nM T35734 CBE64U 76310542 IC50 = 3.1 nM T35734 C7SVJ5 76310543 IC50 = 14.2 nM T35734 CY5FV6 76310544 IC50 = 15.8 nM T35734 C2K5JQ 76310545 IC50 = 29.8 nM T35734 CI7F6E 76310546 IC50 > 100 nM T35734 CX2OW8 76310547 IC50 > 100 nM T35734 C1A8QH 76313824 IC50 = 408 nM T35734 C63UGS 76313825 IC50 = 190 nM T35734 CZ2YQ8 76313826 IC50 = 69 nM T35734 C7YUI4 76317349 IC50 > 10000 nM T35734 CG4YN2 76317350 IC50 = 838 nM T35734 C4U8HZ 76317351 IC50 = 204 nM T35734 CHJ97V 76317352 IC50 = 6.6 nM T35734 CU7I2Z 76317760 IC50 = 2.1 nM T35734 C0EFD4 76321067 IC50 = 4400 nM T35734 C3E4BZ 76321068 IC50 = 3200 nM T35734 C0YSI1 76321069 IC50 > 10000 nM T35734 C2MB7H 76321070 IC50 = 280 nM T35734 C57UCR 76321466 IC50 = 3.3 nM T35734 C7AQ0F 76321467 IC50 = 2.6 nM T35734 C57VPS 76322009 IC50 = 12000 nM T35734 CKFR30 76324719 IC50 = 1500 nM T35734 C4C0RG 76324720 IC50 > 10000 nM T35734 CMC1O9 76325071 IC50 = 8.9 nM T35734 C07MBP 76325072 IC50 = 7.4 nM T35734 CJSG34 76325073 IC50 = 14.7 nM T35734 C9I1AU 76325074 IC50 = 10.7 nM T35734 CW80XU 76325075 IC50 = 12 nM T35734 CS64RF 76325076 IC50 = 18 nM T35734 C1NHT5 76325077 IC50 = 25.2 nM T35734 CGZW93 76325078 IC50 = 26.7 nM T35734 C0SQH2 76325079 IC50 = 2 nM T35734 CN8MZ5 76325631 IC50 > 33000 nM T35734 C7A9ST 76328271 IC50 = 35 nM T35734 C54UPW 76328642 IC50 = 12 nM T35734 C0B8DS 76328643 IC50 = 22.4 nM T35734 C6OHJ5 76328644 IC50 = 4.3 nM T35734 CH2WZ0 76331903 IC50 = 170 nM T35734 C72GIA 76331952 IC50 > 10000 nM T35734 CU7YC0 76331953 IC50 > 10000 nM T35734 C6FUV8 76331954 IC50 > 1000 nM T35734 CQ7AT3 76331955 IC50 = 19 nM T35734 CXU64P 76331956 IC50 = 19 nM T35734 CSUE64 76332318 IC50 = 43.2 nM T35734 C2MS7K 76332319 IC50 = 27.4 nM T35734 C41FLN 76332320 IC50 = 24.4 nM T35734 CAYW74 76332321 IC50 = 94.2 nM T35734 C1RUT0 76332322 IC50 = 27.1 nM T35734 C0NDJ9 76335531 IC50 = 7.9 nM T35734 CQ38GE 76335533 IC50 = 2300 nM T35734 CL1F8Y 76335534 IC50 = 550 nM T35734 COBU42 76335535 IC50 = 5 nM T35734 CQ93ZX 76335954 IC50 = 11.3 nM T35734 CKT50C 76335955 IC50 = 10.2 nM T35734 CRA98Y 76335956 IC50 = 30.3 nM T35734 CLY2O4 84422330 IC50 = 1900 nM T35734 CJY2M4 84425006 IC50 = 4600 nM T35734 CRPT75 90074661 IC50 = 7 nM T35734 CI8V5G 90654760 IC50 = 23810 nM T35734 CV19PA 90654761 IC50 = 47360 nM T35734 C6BZ7A 90654762 IC50 > 50000 nM T35734 CQWY57 90656028 IC50 = 179.2 nM T35734 C13SXH 90656029 IC50 = 26.3 nM T35734 C2KQG0 90656030 IC50 = 7.3 nM T35734 CVCP06 90656031 IC50 = 779.6 nM T35734 C5R3MD 90656032 IC50 = 39.7 nM T35734 CCG50A 90656033 IC50 = 7.2 nM T35734 C83EWU 90656034 IC50 = 2.5 nM T35734 CVS72O 90656035 IC50 = 2.3 nM T35734 CTG69M 90656036 IC50 = 997 nM T35734 COP9T2 90656037 IC50 = 0.8 nM T35734 C0S7GI 90656038 IC50 = 1440 nM T35734 CS80DZ 90656039 IC50 = 161 nM T35734 CEY1W5 90656040 IC50 = 10.4 nM T35734 CX4L3O 90656041 Ki = 2.4 nM T35734 C4NPR7 90668279 IC50 = 77.3 nM T35734 CFI83M 90668280 IC50 = 44.7 nM T35734 CNA84L 90668281 IC50 = 18.8 nM T35734 C53JAL 90668282 IC50 = 321 nM T35734 CX1PD5 90668283 IC50 = 0.6 nM T35734 C9YTX2 90668284 IC50 = 0.4 nM T35734 C8AP1X 90668285 IC50 = 0.5 nM T35734 C5NWD8 91667424 IC50 = 2.3 nM T35734 CPND47 91754971 IC50 = 20 nM T35734 C4EG9D 91754984 IC50 = 20 nM T35734 CEA25K 91754985 IC50 = 13100 nM T35734 CP87IC 91754987 IC50 = 3280 nM T35734 C9BSK6 91754988 IC50 = 180 nM T35734 C2WDJ9 91754989 IC50 = 1320 nM T35734 C4OI8Q 91754990 IC50 = 110 nM T35734 C6R2WN 91754991 IC50 = 1820 nM T35734 CBV1D3 93534208 IC50 = 63 nM T35734 CB2RS8 94519439 IC50 = 44 nM T35734 CD5L1R 94519440 IC50 = 1730 nM T35734 C8ZT0Q 100936503 IC50 = 24000 nM T35734 CBLO69 101403646 IC50 = 18500 nM T35734 C42LCF 102034966 IC50 = 97.6 nM T35734 CF2N5U 102332233 IC50 = 6400 nM T35734 C4EZN8 102369407 IC50 > 500 nM T35734 C1P2HC 105534625 IC50 = 120 nM T35734 CYN18Q 108884731 IC50 = 18500 nM T35734 C5H4JX 108933742 IC50 = 660 nM T35734 CI62TQ 110784491 IC50 = 1200 nM T35734 C05LOZ 118712047 Ki = 0.02 nM T35734 C91AVW 118712048 Ki = 0.23 nM T35734 CVL5X6 118712049 Ki = 111 nM T35734 CREC08 118712050 Ki = 11.2 nM T35734 C5LA9P 118712051 Ki < 0.02 nM T35734 CXRH70 118728601 IC50 = 19.1 nM T35734 C50IFB 118728602 IC50 > 100 nM T35734 CFU3E7 118728603 IC50 = 12 nM T35734 C9ADU1 118728604 IC50 = 75.7 nM T35734 CT2MF1 118728605 IC50 = 2.1 nM T35734 CGI24F 118728606 IC50 = 1.8 nM T35734 C0UM6F 118728607 IC50 = 14.4 nM T35734 C9RDY5 118728608 IC50 = 1.4 nM T35734 CBS14X 118728609 IC50 = 0.7 nM T35734 CP5R8D 118902251 IC50 = 2 nM T35734 CDX21P 119025613 IC50 = 7500 nM T35734 C82VWL 119025614 IC50 = 8600 nM T35734 C0F3PE 119313998 IC50 = 370 nM T35734 C10ESB 122190707 Ki = 200 nM T35734 CU50YN 122190708 Ki = 800 nM T35734 CA9QT1 122190709 Ki = 10400 nM T35734 CK72QZ 122190710 IC50 = 4100 nM T35734 C4FC9O 122193432 IC50 = 120 nM T35734 CGR97Z 122193744 IC50 = 69 nM T35734 CRBY12 122193745 IC50 = 5.1 nM T35734 CGEP51 122193746 IC50 = 30 nM T35734 CC3BH2 122193747 IC50 = 3.8 nM T35734 C1SD3H 122193748 IC50 = 1.7 nM T35734 C8EX3W 122193749 IC50 = 3 nM T35734 CGLD04 122193750 IC50 = 1.8 nM T35734 C45JPS 122193751 IC50 = 2.6 nM T35734 CC8AM7 122193989 IC50 = 17 nM T35734 C64FBZ 122193990 IC50 = 37 nM T35734 CAW20F 122193991 IC50 = 8.2 nM T35734 CR8WP0 122193992 IC50 = 43 nM T35734 CBZU65 122193993 IC50 > 1000 nM T35734 C4WN9I 122195455 IC50 = 15.4 nM T35734 C6BZN5 122195456 IC50 = 12.9 nM T35734 CF0YL3 122195457 IC50 = 4.9 nM T35734 C0F3XD 122195458 IC50 = 29.4 nM T35734 C4SW2H 122195459 IC50 = 44.6 nM T35734 C8X5HV 122195460 IC50 = 16.6 nM T35734 CX70PZ 122195461 IC50 = 10.5 nM T35734 C35UNW 122195462 IC50 = 575.8 nM T35734 CT3XH2 122195463 IC50 = 524.3 nM T35734 C2ETK1 122195464 IC50 = 247.2 nM T35734 C1U2NQ 122195465 IC50 = 190.6 nM T35734 C6G7DJ 122195466 IC50 = 91 nM T35734 CE09BV 122195467 IC50 = 25.8 nM T35734 CLJE23 122195468 IC50 = 15 nM T35734 CC3EK7 122195469 IC50 = 4.1 nM T35734 CJC9A8 122195470 IC50 = 123 nM T35734 CLFG37 122195471 IC50 = 17 nM T35734 CEW86O 122196300 IC50 = 35700 nM T35734 CK37CW 122196301 Ki = 600 nM T35734 C9G8NW 123553842 IC50 = 3 nM T35734 C4RP2D 127038538 IC50 = 2200 nM T35734 CZ41FM 127039679 IC50 = 3800 nM T35734 CF18OQ 127039681 IC50 = 4000 nM T35734 CG1S6F 127039682 IC50 = 30 nM T35734 CXGT91 127039861 IC50 = 1700 nM T35734 CXC23N 127040017 IC50 = 900 nM T35734 C2DMQ6 127040580 IC50 = 70 nM T35734 C6C1TE 127040581 IC50 = 80 nM T35734 CWSN58 127040582 IC50 = 63 nM T35734 C8VXT4 127040583 IC50 = 44 nM T35734 C7XV1H 127040584 IC50 = 1600 nM T35734 CVQT15 127040585 IC50 = 120 nM T35734 C6FC4D 127040586 IC50 = 40 nM T35734 C02ADV 127040870 IC50 = 170 nM T35734 C96SZT 127040871 IC50 = 1000 nM T35734 C9CS8Z 127041189 IC50 = 5000 nM T35734 CN45YE 127041516 IC50 = 570 nM T35734 CH9WU6 127041522 IC50 = 27 nM T35734 C39LHD 127041523 IC50 = 900 nM T35734 CQMD26 127041524 IC50 = 400 nM T35734 CZK7B9 127041525 IC50 = 110 nM T35734 C8IOP5 127041820 IC50 = 9000 nM T35734 C8ZQT1 127041821 IC50 = 250 nM T35734 C3B6SN 127041822 IC50 = 8000 nM T35734 C82RIP 127042123 IC50 = 7200 nM T35734 C9H3DO 127042124 IC50 = 900 nM T35734 C54WUI 127042144 IC50 = 12000 nM T35734 C3I1BC 127042145 IC50 = 120 nM T35734 COUD73 127042146 IC50 = 1200 nM T35734 CRN48C 127042147 IC50 = 30 nM T35734 C74HEQ 127042148 IC50 = 330 nM T35734 C10ZDF 127042456 IC50 = 14000 nM T35734 CU5J1F 127042457 IC50 = 620 nM T35734 C3SFH0 127042459 IC50 = 1500 nM T35734 C40UWZ 127042480 IC50 = 170 nM T35734 C3X0VB 127042481 IC50 = 5000 nM T35734 C1RZE5 127042482 IC50 = 120 nM T35734 C9I0GA 127042483 IC50 = 2500 nM T35734 C8CL0V 127042484 IC50 = 5500 nM T35734 CAC1X8 127042485 IC50 = 8500 nM T35734 CH79WO 127044774 IC50 = 2740 nM T35734 CFUL98 127044775 IC50 = 182 nM T35734 CKU6P0 127044776 IC50 = 302 nM T35734 C7FQG5 127044926 IC50 = 36 nM T35734 C5KZC1 127044927 IC50 = 4500 nM T35734 CZU74Y 127044928 IC50 = 43 nM T35734 CLV54I 127044929 IC50 = 364 nM T35734 CZ5R4K 127044930 IC50 = 65 nM T35734 CGSL16 127044931 IC50 = 22 nM T35734 CC89QV 127045081 IC50 = 19990 nM T35734 C2TYR6 127045089 IC50 = 22 nM T35734 CMS61B 127045090 IC50 = 2030 nM T35734 CI1MP4 127048366 IC50 = 27 nM T35734 CVMU30 127048367 IC50 = 850 nM T35734 CU5E0W 127051507 IC50 = 64 nM T35734 CHU9C7 127051534 IC50 = 1300 nM T35734 CL3M2Y 127051846 IC50 = 300 nM T35734 CG1RN9 127051847 IC50 = 1200 nM T35734 C4WNG7 127052228 IC50 = 7700 nM T35734 CAN02O 127052474 IC50 = 570 nM T35734 CP0S4W 127052475 IC50 = 40 nM T35734 CBY92R 127052476 IC50 = 23 nM T35734 CC7RB8 127052763 IC50 = 75 nM T35734 C4F5VE 127052764 IC50 = 27 nM T35734 C75HWZ 127052765 IC50 = 2500 nM T35734 CIZO79 127068002 IC50 = 60.3 nM T35734 CL15OC 127116223 IC50 = 2050 nM T35734 CO7JB6 130211534 IC50 = 18 nM T35734 C74FUW 130431462 IC50 = 5 nM T35734 C1ZP4G 130431469 IC50 = 2 nM T35734 C6PGV8 130431471 IC50 = 4 nM T35734 C2CZ8L 130431473 IC50 = 2 nM T35734 CMA35H 130431481 IC50 = 3 nM T35734 CC20NA 130431485 IC50 = 5 nM T35734 CFI65G 130431510 IC50 = 3 nM T35734 CQH78B 130431516 IC50 = 2 nM T35734 CE0ZN8 130451190 IC50 = 15 nM T35734 C4NEQ0 130451194 IC50 = 3 nM T35734 C79QKD 130451195 IC50 = 4 nM T35734 CAP96O 130451299 IC50 = 30 nM T35734 CQ27FJ 130451300 IC50 = 4 nM T35734 CW2CG8 131972553 IC50 = 21.1 nM T35734 CS86JX 132487951 IC50 = 400 nM T35734 CAR87V 132487953 IC50 = 14600 nM T35734 CW8LM6 132487954 IC50 = 10700 nM T35734 CKNL89 133081968 IC50 = 2.1 nM T35734 CF65AU 135385301 IC50 = 40 nM T35734 C7O6NY 135393726 IC50 = 148 nM T35734 CWOG26 135393727 IC50 = 160 nM T35734 CQLN71 135393728 IC50 = 58 nM T35734 C5AZX8 136035742 IC50 = 65 nM T35734 C3KG2U 137349604 IC50 = 7050 nM T35734 CG7PY3 137362029 IC50 = 0.4 nM T35734 C8NP6G 137362035 IC50 = 2.9 nM T35734 C5UY1T 137362043 IC50 = 15 nM T35734 CJ45FR 137362044 IC50 = 7 nM T35734 C2RY4M 137362070 IC50 = 13 nM T35734 CJW65C 137362073 IC50 = 2 nM T35734 C70YAR 137362074 IC50 = 2.8 nM T35734 CJ92TM 137362109 IC50 = 3 nM T35734 C4AN6T 137362124 IC50 = 44 nM T35734 C9F6DV 137362127 IC50 = 3.7 nM T35734 CY5PT7 137362372 IC50 = 1.5 nM T35734 CYH0A1 137362374 IC50 = 4 nM T35734 CWI63S 137362887 IC50 = 0.4 nM T35734 CLE03H 137362889 IC50 = 109 nM T35734 CZK87D 137363359 IC50 = 1 nM T35734 C5W7LD 137363713 IC50 = 180 nM T35734 C9R8AG 137363716 IC50 = 190 nM T35734 CAD2P3 137631891 IC50 = 1 nM T35734 CFV9Q1 137633520 IC50 = 1300 nM T35734 C93VAE 137634162 IC50 = 12700 nM T35734 CZ3WM6 137634192 IC50 = 5040 nM T35734 CKL1B0 137636686 IC50 = 18200 nM T35734 CR37SG 137637968 IC50 = 1430 nM T35734 CX3W4Q 137639938 IC50 = 1630 nM T35734 CU04TI 137640615 IC50 = 1.7 nM T35734 C2F6GZ 137640822 IC50 = 390 nM T35734 C39SQB 137641372 IC50 = 170 nM T35734 C2J8BG 137641922 IC50 = 800 nM T35734 C72NWG 137644140 IC50 = 8.9 nM T35734 CS96PL 137644758 IC50 = 510 nM T35734 C09BNW 137645124 IC50 = 910 nM T35734 CS3M4I 137647530 IC50 = 220 nM T35734 CBS06O 137651853 IC50 = 680 nM T35734 CG7B2M 137652547 IC50 = 157 nM T35734 C7MV8K 137653251 IC50 = 19000 nM T35734 CK7JD5 137653822 IC50 = 10000 nM T35734 CF3N9H 137654427 IC50 = 220 nM T35734 C70WUN 137655766 IC50 = 20000 nM T35734 CP9UJ4 137656136 IC50 = 137 nM T35734 C43HUX 137656636 IC50 = 20300 nM T35734 C4IN0L 137658784 IC50 = 1120 nM T35734 CEB57N 137660863 IC50 = 0.6 nM T35734 CSH73J 138756786 IC50 = 3600 nM T35734 CX0L1A 139035063 IC50 = 4000 nM T35734 CR3H2Q 145315259 IC50 = 6 nM T35734 C9XGA5 145955168 IC50 = 7.7 nM T35734 CVPT49 145960364 IC50 = 1248 nM T35734 CXU68C 145960390 IC50 = 987.4 nM T35734 CI42WE 145960483 IC50 = 20.8 nM T35734 CCOS43 145960512 IC50 = 2479 nM T35734 CB68XE 145960691 IC50 = 5334 nM T35734 C5VQ4F 145961058 IC50 = 15.3 nM T35734 C9KIA0 145961401 IC50 = 50248 nM T35734 CAM1B7 145961781 IC50 = 7.2 nM T35734 CT1QG4 145961905 IC50 = 16.1 nM T35734 CEH63N 145961929 IC50 = 14.8 nM T35734 CNF1X4 145962024 IC50 = 5903 nM T35734 C6GO0D 145962103 IC50 = 902 nM T35734 CP06RQ 145962302 IC50 = 152 nM T35734 CV24FB 145962391 IC50 = 216 nM T35734 C1SAK3 145962464 IC50 = 5936 nM T35734 CG8U7A 145962586 IC50 = 57393 nM T35734 C29TRE 145962612 IC50 = 259 nM T35734 CYOF27 145962686 IC50 = 9.8 nM T35734 COZ8P5 145963089 IC50 = 7784 nM T35734 CSA25G 145963092 IC50 = 58 nM T35734 C2NFL3 145963401 IC50 = 90.8 nM T35734 CA5D0U 145963421 IC50 = 52 nM T35734 C41MUS 145963605 IC50 = 15314 nM T35734 CG23SO 145964164 IC50 = 1.82 nM T35734 C6C1ZS 145965196 IC50 = 2.22 nM T35734 CNI29A 145965314 IC50 = 4400 nM T35734 CP7G5E 145966093 IC50 = 0.48 nM T35734 CU6RB2 145972636 IC50 = 0.48 nM T35734 C7JH8Q 145973195 IC50 = 0.96 nM T35734 C46OQL 145975256 IC50 = 8 nM T35734 C07QTF 145975345 IC50 = 1.22 nM T35734 C06JVR 145976112 IC50 = 2 nM T35734 C19QSH 145977289 IC50 = 1.92 nM T35734 C5IA9S 145977816 IC50 > 10000 nM T35734 C6T0ML 145978702 IC50 = 60900 nM T35734 CJV9X0 145979073 IC50 = 1100 nM T35734 C0H2YI 145979664 IC50 = 7000 nM T35734 CY0AQ6 145981186 IC50 = 14 nM T35734 CLCW94 145981341 IC50 = 300 nM T35734 C7V8GI 145987301 IC50 = 410 nM T35734 CVDF45 145987347 IC50 = 680 nM T35734 CL68BS 145992231 IC50 = 550 nM T35734 CI86HD 145992748 IC50 = 150 nM T35734 CK5QF7 145994218 IC50 = 1490 nM T35734 CEU9N6 148483514 IC50 = 8.6 nM T35734 C7FMD1 155513489 IC50 = 5600 nM T35734 CO0GN6 155514213 IC50 = 11.7 nM T35734 C8OGV6 155514713 IC50 = 800 nM T35734 C8Z3YJ 155517011 IC50 = 27200 nM T35734 C5B2IR 155518737 IC50 = 1499.5 nM T35734 CJN65T 155519575 IC50 = 13.9 nM T35734 CWRP89 155519890 IC50 = 21.7 nM T35734 C1NQ4X 155520241 IC50 = 0.5 nM T35734 C9IPA6 155520469 IC50 = 3.2 nM T35734 CJPY40 155521682 IC50 = 1700 nM T35734 C5OV4U 155523230 IC50 = 290 nM T35734 CM1Z7V 155523639 IC50 = 0.4 nM T35734 C7BC2H 155525137 IC50 = 15.2 nM T35734 C7OW9F 155526507 IC50 = 3.3 nM T35734 C01EFS 155528719 IC50 = 1800 nM T35734 CX41BV 155529761 IC50 = 8 nM T35734 C24KXE 155530411 IC50 = 20 nM T35734 CF6AC7 155530648 IC50 = 27500 nM T35734 CT7W5G 155531871 IC50 = 7.2 nM T35734 C5C7PV 155532437 IC50 = 6.5 nM T35734 C2UW0O 155532784 IC50 = 0.6 nM T35734 CH65JO 155533037 IC50 = 35.1 nM T35734 CTH8F2 155534569 IC50 = 25.9 nM T35734 CQF20U 155535260 IC50 = 130 nM T35734 C3S7VL 155537100 IC50 = 4.1 nM T35734 C5PG2L 155537652 IC50 = 740 nM T35734 CA2V8K 155537914 IC50 = 500 nM T35734 CAVL53 155539161 IC50 = 5.2 nM T35734 CAX76U 155540179 IC50 = 6.5 nM T35734 C1YVI3 155542516 IC50 = 18000 nM T35734 CR9S6O 155542667 IC50 = 278.9 nM T35734 CK5H3F 155545531 IC50 = 61.9 nM T35734 C6D0IZ 155545668 IC50 = 300 nM T35734 C9UO2J 155546182 IC50 = 900 nM T35734 C72FXA 155546214 IC50 = 3.4 nM T35734 CQ37FM 155547570 IC50 = 0.5 nM T35734 CJES98 155548156 IC50 = 500 nM T35734 CRW78E 155548442 IC50 = 22500 nM T35734 CHE69M 155553765 IC50 = 600 nM T35734 C24EVD 155554682 IC50 = 100 nM T35734 C3QT0N 155558153 IC50 = 0.8 nM T35734 CL8M9D 155561122 IC50 = 77 nM T35734 CSB69O 155562385 IC50 = 10.3 nM T35734 CED94J 155563098 IC50 = 20100 nM T35734 CVY1U7 155564021 IC50 = 1100 nM T35734 C72LZA 155564090 IC50 = 25.2 nM T35734 C10XMH 155564211 IC50 = 400 nM T35734 CO0KU6 155565005 IC50 = 9.1 nM T35734 CGZ14A 155566111 IC50 = 2 nM T35734 COK1W3 155567033 IC50 = 111.5 nM T35734 D00CHD 44235171 IC50 = 79 nM T35734 D00HAZ 45484885 IC50 = 840 nM T35734 D00RST 9927748 IC50 = 3.7 nM T35734 D00VZE 5029871 IC50 = 2 nM T35734 D01CGC 44235172 IC50 = 11194 nM T35734 D01DZF 5193384 IC50 = 7.9 nM T35734 D01JJV 22932424 IC50 = 28 nM T35734 D01NFH 47379736 IC50 = 12 nM T35734 D01OZF 25014697 IC50 = 39 nM T35734 D02ATA 44235634 IC50 = 8110 nM T35734 D02CKF 44234911 IC50 = 43 nM T35734 D02UJV 25015710 IC50 = 38 nM T35734 D02YEE 45487805 IC50 = 1200 nM T35734 D03CSL 44234662 IC50 = 3480 nM T35734 D03IVU 45267095 IC50 = 152 nM T35734 D04ARH 49782570 IC50 = 3.2 nM T35734 D04NJC 3545369 IC50 = 14 nM T35734 D04PNC 1121089 IC50 = 4000 nM T35734 D05IKY 44235175 IC50 = 66 nM T35734 D05JKG 68770 IC50 = 2800 nM T35734 D05MAT 2235217 IC50 = 746 nM T35734 D05MTA 11417158 IC50 = 1.2 nM T35734 D05NZH 11160856 IC50 = 6200 nM T35734 D06DZO 5071820 IC50 = 159 nM T35734 D06OFY 44582486 IC50 = 392 nM T35734 D06RJQ 11255879 IC50 = 3100 nM T35734 D06WAL 6072 IC50 = 41720 nM T35734 D07BJC 44235174 IC50 = 272 nM T35734 D07BQN 11976254 IC50 = 31 nM T35734 D07HSQ 44419692 IC50 = 100 nM T35734 D07HWV 44235412 IC50 = 7147 nM T35734 D07QNN 82500 IC50 = 14000 nM T35734 D07TOI 11186744 IC50 = 170 nM T35734 D07UIO 44234663 IC50 = 48.5 nM T35734 D08AKP 44235173 IC50 = 10712 nM T35734 D08AZT 22932333 IC50 = 139 nM T35734 D08BFU 5282102 IC50 > 50000 nM T35734 D08HUX 3530525 IC50 = 7 nM T35734 D08IBD 11379743 IC50 = 2100 nM T35734 D08RFH 16756626 IC50 = 2.5 nM T35734 D08RPW 742677 IC50 = 160 nM T35734 D08TWI 44234914 IC50 = 16 nM T35734 D08USX 44475209 IC50 = 120 nM T35734 D08WHU 44582456 IC50 = 1411 nM T35734 D08XYV 44235414 IC50 = 1355 nM T35734 D08YJF 880922 IC50 = 16000 nM T35734 D09ALJ 5280805 IC50 = 24300 nM T35734 D09BUG 10207 IC50 = 26800 nM T35734 D09DPC 17375075 IC50 = 8544 nM T35734 D09FEC 3397178 IC50 = 230 nM T35734 D09VSL 14322900 IC50 = 4200 nM T35734 D09WQW 6420120 IC50 > 100000 nM T35734 D0A1CM 5281855 IC50 = 20700 nM T35734 D0A4VS 16756389 IC50 = 3.9 nM T35734 D0AT6Z 44234916 IC50 = 2596 nM T35734 D0B0ES 751320 IC50 = 190 nM T35734 D0B0MU 44234917 IC50 = 1374 nM T35734 D0B3GP 45487830 IC50 = 520 nM T35734 D0B4CV 4149241 IC50 > 500000 nM T35734 D0BI0Z 11976417 IC50 = 45 nM T35734 D0C1EP 45484883 IC50 = 960 nM T35734 D0C5GW 13451 IC50 = 760 nM T35734 D0C8HN 44234660 IC50 = 770 nM T35734 D0D0KT 4648643 IC50 = 700 nM T35734 D0D3GF 24849868 IC50 = 1200 nM T35734 D0D7ID 4359 IC50 = 140 nM T35734 D0F3PF 2955557 IC50 = 10 nM T35734 D0F3VZ 49782569 IC50 = 3.9 nM T35734 D0F5XQ 16756510 IC50 = 153 nM T35734 D0G8HM 4357 IC50 = 140 nM T35734 D0HC9P 5488619 IC50 = 27430 nM T35734 D0I0YE 1220236 IC50 = 5.1 nM T35734 D0I4KB 49782799 IC50 = 43 nM T35734 D0IC8U 24849867 IC50 = 810 nM T35734 D0IM1Q 45484855 IC50 = 170 nM T35734 D0J0YB 263942 IC50 = 482 nM T35734 D0J5KK 3221297 IC50 = 300 nM T35734 D0J7FK 43608139 IC50 = 3200 nM T35734 D0K6GX 288831 IC50 = 1400 nM T35734 D0K6IW 11976535 IC50 = 8 nM T35734 D0K6OL 880925 IC50 = 6200 nM T35734 D0M0KA 23631476 IC50 = 4.1 nM T35734 D0N1SE 49782798 IC50 = 40 nM T35734 D0NH1E 1383884 IC50 = 1100 nM T35734 D0P3WB 11976309 IC50 = 9.1 nM T35734 D0P8MM 49782797 IC50 = 1700 nM T35734 D0Q8NE 28787671 IC50 = 24 nM T35734 D0R1YP 11644572 IC50 = 1400 nM T35734 D0R6CW 47379737 IC50 = 130 nM T35734 D0RK4K 44582455 IC50 = 365 nM T35734 D0RX9W 4277 IC50 = 25.3 nM T35734 D0S0SH 10069117 IC50 = 0.6 nM T35734 D0S3KS 729989 IC50 = 4800 nM T35734 D0T9ZN 11772500 IC50 = 130 nM T35734 D0TS7G 6420119 IC50 = 36000 nM T35734 D0U0WU 44234656 IC50 = 46 nM T35734 D0U4KM 24849910 IC50 = 2.8 nM T35734 D0U6TM 11382033 IC50 = 100 nM T35734 D0UJ9V 23631733 IC50 = 84 nM T35734 D0V8EQ 44582391 IC50 = 4.7 nM T35734 D0VW6Y 23631475 IC50 = 5.6 nM T35734 D0X1EG 44234912 IC50 = 793 nM T35734 D0X6ZY 11529433 IC50 = 12.6 nM T35734 D0X7IM 7595 IC50 = 390 nM T35734 D0XG0G 11151795 IC50 = 110 nM T35734 D0XS3W 44416958 IC50 = 3800 nM T35734 D0YS1G 23631474 IC50 = 29 nM T35734 D0Z0XL 45484884 IC50 = 1200 nM T35734 D0Z6SS 3090774 IC50 = 17 nM T35734 D0Z8RL 23631734 IC50 = 12 nM T87206 D05EAM 4735 IC50 > 100000 nM T87206 C58UIV 67364 Ki = 5000 nM T87206 CE9P7M 97286 IC50 = 36300 nM T87206 C0L9GX 655480 Ki < 1000 nM T87206 C8SU0E 691392 IC50 = 42100 nM T87206 CFR1V9 3336761 Ki = 17500 nM T87206 CRJ1S6 6486622 Ki = 3600 nM T87206 C0C8FH 28809802 Ki = 25100 nM T03661 D06IAR 60961 Ki = 2180000 nM T03661 D0T3AD 439693 Ki = 0.0001 nM T03661 C1XSZ0 149792 Ki = 122 nM T03661 C7V8HT 149793 Ki = 80 nM T03661 C5CA3B 447342 Ki = 7.7 nM T03661 C5HNK0 448215 Ki = 11 nM T03661 C9UR3Q 448903 Ki = 30 nM T03661 C6Y1IM 449015 Ki = 9.8 nM T03661 C0MHU8 3009363 Ki = 5900 nM T03661 CM86XK 9824827 Ki = 26 nM T03661 CG5L7Z 9842886 IC50 > 100000 nM T03661 CX56JB 10106291 Ki = 40 nM T03661 C81WUI 10173385 IC50 = 8.7 nM T03661 CY6X9U 10238071 IC50 = 8.6 nM T03661 CGQ8F5 10480325 Ki = 4.9 nM T03661 CWPN65 11155059 Ki = 12 nM T03661 CAZ8N1 11164109 Ki = 1300 nM T03661 CU4YM9 11188723 Ki = 6200 nM T03661 CF35KT 11225254 Ki = 34 nM T03661 CWUE05 11225534 Ki = 91 nM T03661 C2T7EK 11235305 Ki = 13 nM T03661 CY5TF2 11294474 Ki = 57 nM T03661 CGQ59M 11350966 Ki = 1900 nM T03661 CG0IL3 11373857 Ki = 17 nM T03661 C30WDR 11394608 Ki = 240 nM T03661 CAN7T5 11403576 Ki = 0.053 nM T03661 CV5FP4 11406877 Ki = 55 nM T03661 CR73FB 11431071 Ki = 38 nM T03661 CC9PM7 11453636 Ki = 17 nM T03661 CTD0L6 11454124 Ki = 13 nM T03661 CF04PG 11774256 Ki = 24 nM T03661 CS4UE8 13989295 Ki = 180000 nM T03661 CI0Y4J 13989301 Ki = 15000 nM T03661 CQ0T3M 16720828 Ki > 10 nM T03661 C3JV8Y 21145345 IC50 = 570 nM T03661 CBYX30 21265683 Ki = 6.3 nM T03661 C6N3VE 22628519 Ki = 54000 nM T03661 CZN72D 24825632 Ki > 100000 nM T03661 C07PUK 24825633 Ki > 100000 nM T03661 C8N6YF 24825634 Ki > 100000 nM T03661 C5PS2M 44272119 Ki = 120 nM T03661 C4IHB8 44327031 Ki = 85000 nM T03661 C03SNC 44344353 Ki = 1200 nM T03661 C6LU7F 46875046 Ki = 0.01 nM T03661 CL0V1B 46875663 Ki = 1410000 nM T03661 COYG70 53318756 Ki = 0.01 nM T03661 CZSC39 53323498 Ki = 0.0025 nM T03661 C6DQ2W 56928836 IC50 = 3700 nM T03661 C2XI3H 71450843 Ki = 0.0025 nM T03661 D03PLV 159738 Ki = 100 nM T03661 D04GWR 447339 IC50 = 700 nM T03661 D08ZMX 449014 Ki = 13 nM T03661 D0D7CM 449013 Ki = 11 nM T03661 D0I6XA 149784 Ki = 0.4 nM T03661 D0L5XY 447340 Ki = 5900 nM T03661 D0R7RB 68368 Ki = 7000 nM T03661 D0T0OW 25447 Ki = 0.0001 nM T03661 D0V4WB 149790 Ki = 2 nM T03661 D0V6TX 447546 Ki = 7.5 nM T75498 D00STL 644241 IC50 = 381 nM T75498 D09EGZ 2719 IC50 = 1500 nM T75498 D0AN7B 896 Ki = 27.6 nM T75498 D0AZ3C 5291 Ki = 39 nM T75498 D0M7JT 216210 IC50 > 10000 nM T75498 D0T1LK 4908 IC50 = 7500 nM T75498 D0WV3U 4893 IC50 = 7.8 nM T75498 D07JTD 132127 IC50 = 126 nM T75498 D0U3EP 445154 Ki = 88 nM T75498 C1LY8B 7019 IC50 = 440 nM T75498 C5JLH9 69088 IC50 > 500000 nM T75498 CF50MK 76137 IC50 = 31100 nM T75498 CO1ED6 96896 IC50 = 11200 nM T75498 C3UA0B 101252 IC50 = 60800 nM T75498 C1U3VY 124075 IC50 = 54100 nM T75498 C0O3TQ 126437 IC50 = 35 nM T75498 CTW6M9 152481 IC50 = 250 nM T75498 CJU01I 152483 IC50 = 170 nM T75498 CQF84T 154480 IC50 = 597 nM T75498 CMZ7A3 195276 IC50 = 13000 nM T75498 CMO0A9 235279 IC50 = 15300 nM T75498 CX1NP4 291622 IC50 = 35500 nM T75498 C3XY9B 372186 IC50 = 11700 nM T75498 CGW28U 408998 IC50 = 68 nM T75498 C6ES5O 432303 IC50 = 50 nM T75498 C5K7DO 438560 IC50 = 1833 nM T75498 CB2GN1 438565 IC50 = 1333 nM T75498 CL67WS 446804 IC50 = 800 nM T75498 CS4C8A 472392 IC50 = 2047 nM T75498 CLZ2C8 625699 IC50 = 36800 nM T75498 CE4JQ8 782123 IC50 = 24100 nM T75498 CO91JY 784729 IC50 = 5500 nM T75498 CBO9W5 906605 IC50 = 41.69 nM T75498 CJY81E 3071630 IC50 = 43.65 nM T75498 C34HKN 3071633 IC50 = 61.66 nM T75498 C4IR7N 3071639 IC50 = 28.84 nM T75498 COT3G9 3956219 Ki = 1000 nM T75498 C23LQS 5284422 IC50 = 640 nM T75498 C9R3TF 5318763 IC50 = 3840 nM T75498 C4G5QC 5387294 IC50 = 37100 nM T75498 CK0U7H 5484463 IC50 = 2700 nM T75498 C0HRE2 5919990 IC50 = 500 nM T75498 C76CYU 9555351 IC50 = 10 nM T75498 CL2YG0 9594974 IC50 = 103 nM T75498 C6MBQ4 9794567 IC50 = 6000 nM T75498 CDW90R 9816335 Ki = 3570 nM T75498 CWG0C2 9817006 IC50 = 37 nM T75498 CLVE32 9841851 Ki = 48 nM T75498 CXO8S2 9859969 IC50 = 18 nM T75498 CIZD48 9860698 Ki = 1550 nM T75498 C05WRO 9861677 IC50 = 18.2 nM T75498 C01BWX 10062381 IC50 = 70.79 nM T75498 CT03BO 10069719 Ki = 0.18 nM T75498 CBS8C3 10092427 IC50 = 0.302 nM T75498 CGTH05 10105780 IC50 = 9300 nM T75498 CSUN05 10454621 IC50 = 0.1288 nM T75498 CQZ4J3 10873443 Ki = 6.1 nM T75498 CQ35SF 10901399 Ki = 785 nM T75498 C72HJV 10912753 Ki = 812 nM T75498 CCM69E 10933826 Ki = 561 nM T75498 CJ52CX 10946222 IC50 = 0.309 nM T75498 C6LKR7 10956792 Ki = 1.1 nM T75498 CLT5I9 10978708 Ki = 5490 nM T75498 CNA63S 10988162 Ki = 4180 nM T75498 C2LMW6 10992102 Ki = 1770 nM T75498 CDL84Z 11000600 Ki = 9.09 nM T75498 CZEM06 11012504 Ki > 10000 nM T75498 C1NS8V 11023001 Ki = 608 nM T75498 C9JSR3 11033951 Ki = 2600 nM T75498 C4KCN5 11033952 Ki = 4580 nM T75498 CLTG23 11044386 Ki = 374 nM T75498 C71CPN 11053973 Ki = 686 nM T75498 CM3IT6 11054448 Ki = 760 nM T75498 C7EAI8 11065731 Ki = 1000 nM T75498 CU18OA 11066559 Ki = 353 nM T75498 CV4J9D 11076229 Ki = 2270 nM T75498 C8GJ3N 11076291 Ki = 782 nM T75498 CT8DG3 11076588 Ki = 428 nM T75498 C8KO9X 11079938 Ki = 70 nM T75498 C3B4EN 11086040 Ki = 1190 nM T75498 CP5HA6 11096503 Ki = 1810 nM T75498 C0MHQ5 11097218 Ki > 10000 nM T75498 C9R2PL 11100761 Ki = 0.088 nM T75498 C8SZ9C 11100842 Ki = 2450 nM T75498 C5ZW2F 11107609 Ki = 48.6 nM T75498 CJ94CS 11117958 Ki = 372 nM T75498 CUN10Q 11129533 Ki = 837 nM T75498 C0L2IW 11414230 IC50 = 4600 nM T75498 CX82FH 11471958 IC50 = 31600 nM T75498 CH2T9J 11681568 IC50 = 59 nM T75498 CDRK23 11770705 Ki = 467 nM T75498 C8LYO7 11776674 Ki = 2.8 nM T75498 CG27TX 11780348 Ki = 3150 nM T75498 CLI54S 11821384 Ki = 2230 nM T75498 C92OWZ 14929519 IC50 > 500000 nM T75498 CQY85F 15523939 Ki = 316 nM T75498 C68TWS 15680107 IC50 = 46 nM T75498 CI19XZ 17956989 IC50 = 56.23 nM T75498 CM1C9Y 17956992 IC50 = 67.61 nM T75498 CWC8V1 17957000 IC50 = 0.39 nM T75498 CXG63C 17957007 IC50 = 22.91 nM T75498 CW7FB8 18007990 IC50 = 7.762 nM T75498 CW69VB 18174981 IC50 = 15.85 nM T75498 CZ2H3M 18175008 IC50 = 32 nM T75498 CE6YD4 18175028 IC50 = 4.9 nM T75498 CX7D3G 18175032 IC50 = 9.1 nM T75498 CNI15A 18175044 IC50 = 14.13 nM T75498 C7ZS9J 18175084 IC50 = 10.96 nM T75498 C24JYE 19577710 IC50 = 519 nM T75498 CQ7M4S 21679909 IC50 = 18200 nM T75498 C6ZQD8 21916760 IC50 = 21 nM T75498 C5QAW8 21996451 Ki = 497 nM T75498 C7PRG0 22922685 Ki = 946 nM T75498 C1T6YF 24721598 IC50 = 13500 nM T75498 CM9JZ7 24803338 IC50 = 97 nM T75498 CU3M5Q 24803501 IC50 = 83 nM T75498 CB0Z9H 25093729 IC50 = 27600 nM T75498 CRQ41A 25113669 IC50 = 61 nM T75498 CF64XU 25242322 IC50 = 20800 nM T75498 C9JF5O 37559937 IC50 = 28.18 nM T75498 C93BZJ 42618027 IC50 = 6200 nM T75498 C4YXR5 42618028 IC50 = 29300 nM T75498 CVLR83 42618034 IC50 > 500000 nM T75498 CUWO14 42618035 IC50 > 500000 nM T75498 CF95VB 44563733 IC50 = 14200 nM T75498 CM7N8F 44563734 IC50 = 12000 nM T75498 C4FZQ3 44563735 IC50 = 20100 nM T75498 C3C9PD 44563736 IC50 = 33700 nM T75498 CI72ZE 44563763 IC50 = 730 nM T75498 C2ZRI1 44563764 IC50 = 6800 nM T75498 CZDV56 44563766 IC50 = 13000 nM T75498 CQ50LO 44563767 IC50 = 39000 nM T75498 CGT24V 44563774 IC50 = 13000 nM T75498 C04FCZ 44563805 IC50 = 2800 nM T75498 CTB3C7 44563806 IC50 = 4800 nM T75498 CYQS75 44563814 IC50 = 180 nM T75498 CRT8Q1 44571459 IC50 = 10900 nM T75498 C8MK4E 44571460 IC50 = 16300 nM T75498 C0QLE1 44581531 IC50 = 61.66 nM T75498 CJVW31 44581532 IC50 = 14.13 nM T75498 C4ISH0 44581533 IC50 = 53.7 nM T75498 C6U7IO 44581534 IC50 = 51.29 nM T75498 CL6FB9 44581569 IC50 = 23.99 nM T75498 C6SND4 44581570 IC50 = 12.02 nM T75498 C8WJS6 44581613 IC50 = 52.48 nM T75498 CD9YN4 44581689 IC50 = 3.02 nM T75498 CR59BF 44593609 IC50 = 67.61 nM T75498 C8S0ZG 44593610 IC50 = 10.96 nM T75498 C4LTW3 45480965 IC50 = 18 nM T75498 C5DNU4 45481036 IC50 = 1420 nM T75498 C9QVR3 46231191 IC50 = 783 nM T75498 C6GC7K 46231192 IC50 = 1483 nM T75498 C86BIK 46231193 IC50 = 517 nM T75498 CKGV86 46231194 IC50 = 483 nM T75498 C5M1NJ 46231195 IC50 = 987 nM T75498 CIVO25 46231242 IC50 = 98 nM T75498 C5GEO9 46231243 IC50 = 427 nM T75498 CKZ83D 46231244 IC50 = 767 nM T75498 CI0F2H 46231245 IC50 = 350 nM T75498 CY0H6O 46231246 IC50 = 567 nM T75498 CMX69C 46231284 IC50 = 98 nM T75498 C1DJV8 46231285 IC50 = 167 nM T75498 CO74HZ 46231286 IC50 = 117 nM T75498 C3G0ME 49855794 IC50 = 186 nM T75498 C5QFJ4 49855795 IC50 = 18500 nM T75498 CB40UI 49855796 IC50 = 690 nM T75498 CFH9S0 49855798 IC50 = 160 nM T75498 CW04BD 49855799 IC50 = 450 nM T75498 C19XQH 49855986 IC50 = 3300 nM T75498 C3DI8U 49855987 IC50 = 320 nM T75498 COIW92 49855988 IC50 = 10500 nM T75498 C7RBG6 49855989 IC50 = 4800 nM T75498 C8WMJ6 49855991 IC50 = 11300 nM T75498 CQ3ON9 49855992 IC50 = 4100 nM T75498 CK52FD 49855993 IC50 = 3500 nM T75498 CJ1ME4 52941605 IC50 = 20000 nM T75498 C8FT4D 52943732 IC50 = 22000 nM T75498 C2JI3P 54757302 IC50 = 74 nM T75498 CIC83T 54757396 IC50 = 14 nM T75498 C85DMY 54757397 IC50 = 73 nM T75498 C1PBZ0 54757398 IC50 = 205 nM T75498 CJ01PA 54757399 IC50 = 97 nM T75498 CNJ94P 54757400 IC50 = 96 nM T75498 C8F1QU 54757401 IC50 = 56 nM T75498 C6D7RQ 54757402 IC50 = 47 nM T75498 CK9S5Y 54757501 IC50 = 42 nM T75498 CP4XC0 54765330 IC50 = 4.1 nM T75498 COW91E 56945975 IC50 = 3300 nM T75498 CALE95 56945976 IC50 = 5600 nM T75498 C64LQD 56945977 IC50 = 1100 nM T75498 C0C3VT 56945978 IC50 > 100000 nM T75498 C6XSK1 56945979 IC50 = 9000 nM T75498 CPN32V 56945980 IC50 = 4000 nM T75498 C43OCV 56945981 IC50 = 1600 nM T75498 C5JD2S 56946077 IC50 = 1500 nM T75498 C5Y0FB 56946078 IC50 = 1800 nM T75498 C4XTE7 56946079 IC50 = 240 nM T75498 CKG1J2 56946080 IC50 = 150 nM T75498 CPT0H4 56946082 IC50 = 22100 nM T75498 CJ3O9T 56946085 IC50 = 5800 nM T75498 CSW1G8 56946186 IC50 = 7800 nM T75498 CO0EX9 56946187 IC50 = 25200 nM T75498 CAHD15 69641392 IC50 = 16800 nM T75498 CNZ05C 71452564 IC50 = 14100 nM T75498 CU5B2I 71452565 IC50 = 200 nM T75498 C86DPV 71459796 IC50 = 20700 nM T75498 C3HM5I 71463252 IC50 = 7000 nM T75498 CA2I7D 72164104 IC50 = 5900 nM T75498 CY81HD 72164105 IC50 = 25500 nM T75498 CN4HM9 72164106 IC50 = 5100 nM T75498 CMNK94 72164222 IC50 = 24200 nM T75498 C8HK1W 72164225 IC50 = 27500 nM T75498 CET9B4 72164348 IC50 = 9300 nM T75498 C40STG 73350847 IC50 = 9900 nM T75498 CBY19W 73353800 IC50 = 5500 nM T75498 C8XH4M 73355326 IC50 = 6700 nM T75498 C1HLV4 127025379 IC50 = 35 nM T75498 C5RA7Q 127026859 IC50 = 202 nM T75498 CE3UI7 127027830 IC50 = 98 nM T75498 C5Q6HL 127027832 IC50 = 505 nM T75498 CAK10X 127027834 IC50 = 27 nM T75498 CZPH42 127027836 IC50 = 141 nM T75498 CHXK80 127027837 IC50 = 72 nM T75498 C8Q0HD 127027839 IC50 = 509.9 nM T75498 C6TX2R 127027840 IC50 = 14.5 nM T75498 C59MKW 127027841 IC50 = 24 nM T75498 C4EH2F 127027842 IC50 = 832 nM T75498 CHR1N6 127027843 IC50 = 410 nM T75498 CKGV24 127028432 IC50 = 140 nM T75498 CD3MH9 135468602 IC50 = 13 nM T75498 C3U5YT 136025850 IC50 = 2900 nM T75498 CTNU40 136026141 IC50 = 1400 nM T75498 CK6LZ7 136059932 IC50 = 480 nM T75498 CR5F0A 136086891 IC50 = 26900 nM T75498 CBOT34 137644672 IC50 = 4500 nM T75498 CCT9E0 137649044 IC50 = 5100 nM T75498 CX91TG 137651399 IC50 = 63000 nM T75498 C64WJE 137655331 IC50 = 19000 nM T75498 C73IOA 145968145 IC50 = 2000 nM T75498 C7UHQ9 145968667 IC50 = 1140 nM T75498 C4RV2G 145969476 IC50 = 773 nM T75498 C3ORP6 145970380 IC50 = 1111 nM T75498 C9DTO4 155510881 IC50 = 15 nM T75498 C30PXS 155512198 IC50 = 55 nM T75498 C18QLG 155516641 IC50 = 70 nM T75498 CC92QZ 155516868 IC50 = 90 nM T75498 C6Y5NF 155519545 IC50 = 2906 nM T75498 CY2WZ9 155523643 IC50 = 372 nM T75498 CAYE51 155529896 IC50 = 40 nM T75498 C26PCQ 155532551 IC50 = 137 nM T75498 CHC9E0 155533203 IC50 = 595 nM T75498 CGK30C 155536913 IC50 > 10000 nM T75498 CY5C3W 155544355 IC50 = 472 nM T75498 C5D1PY 155546729 IC50 = 64 nM T75498 CNK4E7 155549262 IC50 = 125 nM T75498 CH3E1N 155555454 IC50 = 2070 nM T75498 CRX7G1 155557525 IC50 = 550 nM T75498 CJS1D4 155557679 IC50 = 46 nM T75498 D00AII 5281727 IC50 = 5100 nM T75498 D00DSW 6035704 IC50 = 6500 nM T75498 D00GIU 21123062 IC50 = 1900 nM T75498 D00GUG 6305573 IC50 = 9600 nM T75498 D00OTC 5385086 IC50 = 15000 nM T75498 D00SNO 438569 IC50 = 830 nM T75498 D01DYZ 3656761 IC50 = 2700 nM T75498 D01JID 378422 IC50 = 6 nM T75498 D01LAU 4284525 IC50 = 2.7 nM T75498 D01WRT 327137 IC50 = 5000 nM T75498 D01ZKN 438572 IC50 = 172 nM T75498 D02DOX 386223 IC50 = 2900 nM T75498 D02GDG 5466653 IC50 = 3800 nM T75498 D02NED 154479 IC50 = 50 nM T75498 D03GWA 382414 IC50 = 2000 nM T75498 D03QRT 438550 IC50 = 1000 nM T75498 D03SBI 378419 IC50 = 99 nM T75498 D04KTJ 438570 IC50 = 323 nM T75498 D04LWL 97252 IC50 = 18200 nM T75498 D04PMX 8601 IC50 = 3300 nM T75498 D04UGI 438571 IC50 = 693 nM T75498 D05GDD 371512 IC50 = 427 nM T75498 D05TZK 15282960 IC50 = 1700 nM T75498 D05YCI 42618032 IC50 = 10000 nM T75498 D05ZUX 44207909 Ki >= 1000 nM T75498 D06CHV 5940197 IC50 = 1800 nM T75498 D06GRP 5864101 IC50 = 3200 nM T75498 D06UQR 15306616 IC50 = 6000 nM T75498 D07OAH 5015534 IC50 = 5500 nM T75498 D08FHU 42618033 IC50 = 7000 nM T75498 D08ISK 42618030 IC50 = 8800 nM T75498 D08NCP 378420 IC50 = 17 nM T75498 D08NWU 378421 IC50 = 31 nM T75498 D08WKQ 5905819 IC50 = 5300 nM T75498 D09DRS 42618031 IC50 = 1900 nM T75498 D09MQF 15696376 IC50 = 270 nM T75498 D09XVU 9569316 IC50 = 6200 nM T75498 D0C8KC 1504717 IC50 = 4100 nM T75498 D0E0DQ 371510 IC50 = 296 nM T75498 D0G7MJ 5934332 IC50 = 6000 nM T75498 D0H3LU 258058 IC50 = 2100 nM T75498 D0H6YF 115348 Ki = 6.5 nM T75498 D0I3PD 373149 IC50 = 3500 nM T75498 D0K0TO 3694504 IC50 = 2100 nM T75498 D0L3AJ 5324988 IC50 = 5800 nM T75498 D0M0WT 264430 IC50 = 6000 nM T75498 D0M7RM 5884626 IC50 = 5800 nM T75498 D0O2GK 10059864 IC50 = 64.57 nM T75498 D0O4YS 42618026 IC50 = 10800 nM T75498 D0O6NU 132128 IC50 = 16 nM T75498 D0O9NE 5388063 IC50 = 14600 nM T75498 D0OT1Z 135502354 IC50 = 1400 nM T75498 D0Q8JE 367850 IC50 = 9 nM T75498 D0Q8UZ 18785180 IC50 = 1700 nM T75498 D0S1AY 269167 IC50 = 10800 nM T75498 D0S6RL 4043484 IC50 = 5100 nM T75498 D0T2RY 9948320 Ki >= 1000 nM T75498 D0T5NO 15306617 IC50 = 10800 nM T75498 D0TT3K 438548 IC50 = 953 nM T75498 D0UB3V 5351382 IC50 = 4900 nM T75498 D0W8VX 4550667 IC50 = 2000 nM T75498 D0W9ZH 52942470 IC50 = 5000 nM T75498 D0WW2D 434764 IC50 = 1800 nM T75498 D0XQ6T 42618029 IC50 = 9300 nM T75498 D0Z9MG 434864 IC50 = 6000 nM T83059 D0J9HW 23725625 IC50 > 3000 nM T83059 C1NOK3 2946601 IC50 = 1230 nM T83059 CG5A7W 16013152 IC50 = 1010 nM T83059 CNI3Y5 44483163 EC50 = 2500 nM T83059 CTE39K 49832752 IC50 = 140 nM T83059 CXR9G1 49833459 IC50 = 420 nM T83059 C9V5PW 49834204 IC50 > 10000 nM T83059 C2TG1V 57378623 IC50 = 6300 nM T83059 CX17EU 57378738 IC50 = 70 nM T83059 C6O1UZ 58829329 IC50 = 2000 nM T83059 CD3HT9 67960134 IC50 = 4.5 nM T83059 CA9VM2 68166499 IC50 > 10000 nM T83059 CR5VF9 68166507 IC50 > 10000 nM T83059 CCL8N3 68166517 IC50 = 3920 nM T83059 C4EIK5 68166523 IC50 = 4530 nM T83059 CWV26A 68166560 IC50 = 50 nM T83059 C7QLY3 71464718 IC50 = 2100 nM T83059 CED5V6 71622125 IC50 = 380 nM T83059 CI0GU8 71660496 EC50 = 52 nM T83059 CI98LH 71680701 IC50 = 7300 nM T83059 CHOZ71 71680703 EC50 > 25000 nM T83059 CL20JN 71680704 EC50 > 25000 nM T83059 CBH64M 71680705 IC50 = 1100 nM T83059 C91BGF 71680860 IC50 = 4000 nM T83059 COP6V9 71680863 EC50 = 1010 nM T83059 CBS20R 71681023 IC50 = 390 nM T83059 C1KT7H 71681028 IC50 = 200 nM T83059 CH1FS9 71681175 IC50 = 73 nM T83059 CZ1H8S 71681176 EC50 = 190 nM T83059 CCAK12 71681177 IC50 = 140 nM T83059 CHO50K 71681178 EC50 = 2000 nM T83059 CJO9X1 71681179 EC50 = 73 nM T83059 CJ34PZ 71681180 IC50 = 270 nM T83059 C2RGP3 71681329 IC50 = 67 nM T83059 CI5E8F 71681330 EC50 = 61 nM T83059 C32RCL 71681331 IC50 = 170 nM T83059 CVJ86T 71681485 IC50 = 520 nM T83059 CY12QO 71681487 IC50 = 1710 nM T83059 CH4V6D 71681649 EC50 = 390 nM T83059 CFM05A 71683060 EC50 > 25000 nM T83059 C1MP6Q 71683061 IC50 > 10000 nM T83059 C21VJG 71719343 IC50 = 4500 nM T83059 CMC2J4 72193935 IC50 = 233 nM T83059 C2U6AT 72699516 EC50 = 7 nM T83059 C3E9CI 72699517 EC50 = 2 nM T83059 CO4U3W 72699596 EC50 = 810 nM T83059 CR3ZE1 72699600 EC50 = 127 nM T83059 CJP9L5 72699677 EC50 = 320 nM T83059 C8AE1X 72699858 EC50 = 341 nM T83059 CA0X9C 72699953 EC50 = 47 nM T83059 CLQ5E2 72700032 EC50 = 31 nM T83059 C46DHU 72724967 IC50 = 392 nM T83059 CTWE30 73347820 IC50 = 131 nM T83059 CK9X5R 73356483 IC50 = 150 nM T83059 C3XO5D 89649815 IC50 = 360 nM T83059 C83KNV 89661926 IC50 = 690 nM T83059 C2XR5Q 92045137 IC50 = 222 nM T83059 CV0NZ7 105539834 IC50 = 1910 nM T83059 CLZ1U3 118498201 EC50 = 0.26 nM T83059 CT78JM 118498266 EC50 = 0.22 nM T83059 C1VB9L 118507411 EC50 = 2.9 nM T83059 C02SDC 122423373 IC50 > 3000 nM T83059 CF2NO9 127037410 IC50 = 790 nM T83059 C1KBX6 135417551 IC50 = 1536 nM T83059 C1PE8H 135417609 IC50 = 1294 nM T83059 C47LAF 135418940 IC50 = 11 nM T83059 CM5Q1Z 135430309 EC50 > 30000 nM T83059 CH14EB 135443955 EC50 = 1500 nM T83059 C8XI3K 135448518 EC50 > 30000 nM T83059 CU3FW2 135566794 IC50 = 36000 nM T83059 CT1DZ8 135644892 IC50 = 1066 nM T83059 C38XBR 135652704 IC50 = 42.9 nM T83059 C54NVS 136175126 EC50 = 21 nM T83059 CVH7R6 136175127 EC50 = 48 nM T83059 CS5PH8 136175128 EC50 = 1.3 nM T83059 CM4PB2 136236970 EC50 = 614 nM T83059 C50JYC 136236972 EC50 = 620 nM T83059 C1WG3C 136236974 EC50 = 590 nM T83059 CF1H5N 136236975 EC50 = 6300 nM T83059 CU17IT 136236976 EC50 = 1100 nM T83059 C71FDZ 136236977 EC50 = 360 nM T83059 CCL4D6 136236978 EC50 = 760 nM T83059 C9WHB4 136236979 EC50 = 310 nM T83059 C68GON 136236980 EC50 = 700 nM T83059 C18MSY 136236981 EC50 = 319 nM T83059 CF01JX 136236982 EC50 = 456 nM T83059 CYF2I1 136236983 EC50 = 12000 nM T83059 C3ZW8J 136236994 EC50 = 79 nM T83059 CN0J1C 136236995 EC50 = 2000 nM T83059 CHJ8I2 136236997 EC50 = 31 nM T83059 C0LB6W 136236998 EC50 = 37 nM T83059 CVB4D7 136237000 EC50 = 610 nM T83059 CSB3Y1 136237004 EC50 = 170 nM T83059 C4H8ZN 136237010 EC50 = 940 nM T83059 CR07BF 136244504 IC50 = 11 nM T83059 CUPY84 136268378 IC50 = 531 nM T83059 C6T9OI 136947736 EC50 = 50 nM T83059 C91WJF 136947741 EC50 = 53 nM T83059 CFS5Z4 136947743 EC50 = 3900 nM T83059 CVM4S9 136947751 EC50 = 2100 nM T83059 CMN5H6 137169065 IC50 = 832 nM T83059 C4R7VI 137701512 IC50 = 12.1 nM T83059 CWLV03 138594154 IC50 = 6.3 nM T83059 CDW5N1 138594164 IC50 = 0.3 nM T83059 CSK82I 138594166 IC50 = 1.3 nM T83059 CD1M0Y 138594171 IC50 = 3.2 nM T83059 C9QYJ3 138594172 IC50 = 0.1 nM T83059 C1XSH7 138594194 IC50 = 0.3 nM T83059 C4JO9N 138594198 IC50 = 1.6 nM T83059 C7I1CT 138594235 IC50 = 2.7 nM T83059 CVI5N9 138594242 IC50 = 1.1 nM T83059 CS8U3T 138594273 IC50 = 0.3 nM T83059 CYR32Z 138594277 IC50 = 1.1 nM T83059 CNSV30 138594278 IC50 = 0.1 nM T83059 C1C2AS 138594290 IC50 = 2.5 nM T83059 C34OCY 138594292 IC50 = 13.7 nM T83059 CUA1E8 138594320 IC50 = 0.8 nM T83059 CGE6Q5 138594327 IC50 = 0.4 nM T83059 C0RST4 138594360 IC50 = 1347 nM T83059 C4K7MW 138594363 IC50 = 13.9 nM T83059 CNW2O9 138594369 IC50 = 247 nM T83059 C3F7MV 138594378 IC50 = 609 nM T83059 C6YU8S 138594385 IC50 = 454 nM T83059 C48AGS 138594414 IC50 = 352 nM T83059 CA49EZ 138594436 IC50 = 608 nM T83059 CL6EV4 138594465 IC50 = 507 nM T83059 CJL05F 138594467 IC50 = 799 nM T83059 CX4SL6 138594472 IC50 = 72.4 nM T83059 C3E5IU 138594491 IC50 = 4.4 nM T83059 C13EVQ 138594498 IC50 = 342 nM T83059 C4L9XQ 138594506 IC50 = 362 nM T83059 CKF1W3 138594528 IC50 = 623 nM T83059 C98NUR 138594556 IC50 = 4.5 nM T83059 CDZ43N 138594558 IC50 = 14.4 nM T83059 CLD3J5 138594570 IC50 = 0.9 nM T83059 CWVO67 138594578 IC50 = 119 nM T83059 C6QD2W 138594607 IC50 = 21.5 nM T83059 CP6Y5L 138594610 IC50 = 1.5 nM T83059 CSQJ12 138594627 IC50 = 0.2 nM T83059 CEOJ61 138594628 IC50 = 31.1 nM T83059 CU4O9K 138594631 IC50 = 533 nM T83059 C0A4FG 138594645 IC50 = 369 nM T83059 CN3U9X 138594667 IC50 = 19.8 nM T83059 CQK29G 138594732 IC50 = 818 nM T83059 CCU4I1 138594747 IC50 = 43.9 nM T83059 C1KWY7 138594763 IC50 = 91.2 nM T83059 C9HR2J 138594785 IC50 > 10000 nM T83059 CP4NF9 138594790 IC50 = 591 nM T83059 CF74SW 138594809 IC50 = 496 nM T83059 CF7ZR5 138594952 IC50 = 2.1 nM T83059 CW5E6D 138594964 IC50 = 657 nM T83059 CURM89 138594969 IC50 = 52.9 nM T83059 C72QVS 138595093 IC50 = 1605 nM T83059 C8I9CD 142613964 IC50 = 110 nM T83059 CPY72O 153951026 EC50 = 1300 nM T83059 CWV08R 155511996 IC50 = 7282 nM T83059 CZ78CA 155513337 IC50 = 5401 nM T83059 CRX36I 155515281 IC50 = 5.7 nM T83059 CC9J2N 155516254 IC50 = 4.6 nM T83059 C6EJ7I 155518170 IC50 > 10000 nM T83059 CIC9H8 155518184 IC50 = 0.1 nM T83059 C1DL6E 155518640 IC50 = 2246 nM T83059 CGKW04 155520067 IC50 > 10000 nM T83059 CHV6T4 155521523 IC50 = 23.2 nM T83059 CUM52X 155522687 IC50 = 114 nM T83059 CEP6Y5 155528458 IC50 = 1971 nM T83059 C91IPT 155529963 IC50 = 14.5 nM T83059 CA9XP1 155531429 IC50 = 221 nM T83059 CL2PO4 155532179 IC50 = 0.3 nM T83059 C09PYD 155532212 IC50 = 1009 nM T83059 C4JPD1 155532717 IC50 = 0.7 nM T83059 CZL4U1 155534087 IC50 = 0.2 nM T83059 CV2MX1 155535415 IC50 = 1161 nM T83059 CWM48X 155538013 IC50 = 403 nM T83059 CU65VW 155540828 IC50 > 10000 nM T83059 CZN0O1 155541146 IC50 > 10000 nM T83059 C9INM1 155543325 IC50 = 83.9 nM T83059 CO0E8F 155549220 IC50 = 148 nM T83059 CD5C9R 155550189 IC50 > 10000 nM T83059 C4P3QD 155553178 IC50 = 918 nM T83059 CIYH06 155556919 IC50 > 10000 nM T83059 CXAJ25 155557028 IC50 = 36.5 nM T83059 CWH8D0 155561438 IC50 = 7.2 nM T83059 C46UYI 155562058 IC50 = 9144 nM T83059 COH6X1 155564702 IC50 = 36.5 nM T83059 D0T2QL 444539 IC50 = 685 nM T34816 C4AXO5 6539241 Ki = 5000 nM T34816 C98FEY 11285691 Ki = 35 nM T34816 D08AES 11578664 Ki = 478 nM T41580 D01AZG 5073 Ki = 1000 nM T41580 D01JGV 441975 Ki = 14.5 nM T41580 D01JUF 5775 Ki = 7.6 nM T41580 D03MIR 3157 Ki > 5000 nM T41580 D03SKR 2803 Ki = 6.166 nM T41580 D05ZIK 4205 IC50 = 223.87 nM T41580 D06OFS 68712 Ki = 42.66 nM T41580 D07MOX 439260 EC50 = 61.66 nM T41580 D09EBS 4636 Ki = 5370.32 nM T41580 D0AE3X 2435 Ki = 34.67 nM T41580 D0CQ0Z 33630 Ki = 401 nM T41580 D0G8NN 119570 Ki = 67.7 nM T41580 D0H3HM 60795 Ki = 1000 nM T41580 D0H4JM 8969 Ki = 1.16 nM T41580 D0H7KF 5002 Ki = 1000 nM T41580 D0K0MW 30668 Ki = 67.61 nM T41580 D0P9RF 5401 Ki = 26 nM T41580 D0V4QS 135398745 Ki = 100 nM T41580 D0WV3U 4893 Ki = 13 nM T41580 D0Z1RV 135398737 Ki = 100 nM T41580 D05LGX 213041 Ki = 6.761 nM T41580 D0LI1C 44469321 IC50 > 10000 nM T41580 D0N1HW 5311200 Ki = 160 nM T41580 D00OWF 5280953 Ki = 1130 nM T41580 D02LHR 33625 Ki = 528 nM T41580 D03QMR 5685 Ki = 28 nM T41580 D05OVC 71310 Ki = 2.239 nM T41580 D08OWQ 122295 Ki = 142 nM T41580 D0B1MJ 6918097 Ki = 660 nM T41580 D0K9JP 9928332 Ki = 11 nM T41580 D0N7LZ 126225 Ki = 3.4 nM T41580 C5H9CN 9287 Ki > 10000 nM T41580 CL3T5Z 27013 Ki < 100 nM T41580 CU86VK 54459 IC50 = 19.5 nM T41580 C28VFY 60602 Ki = 420 nM T41580 CKR4N3 122065 Ki = 56 nM T41580 C2H1VA 131829 Ki = 48.98 nM T41580 CF4V5Q 185076 Ki = 8.913 nM T41580 CH6WT3 218362 Ki = 2.138 nM T41580 CQ5Z8Y 294234 Ki = 9.772 nM T41580 CAQ2J0 3034396 Ki = 9290 nM T41580 CS2Q1G 3045401 IC50 = 2.57 nM T41580 CU4T6Q 3086326 Ki = 69.18 nM T41580 C3A1FO 6604789 Ki = 3162.28 nM T41580 C8ZBJ9 7059292 Ki = 933.25 nM T41580 C5Z2KM 9805944 Ki = 7 nM T41580 CJ67XC 9815610 Ki = 621 nM T41580 C9PZN8 9815633 Ki = 99 nM T41580 C5A8UR 9815707 Ki = 5.888 nM T41580 CXP87Y 9816063 Ki = 141 nM T41580 C1X0UA 9817256 Ki < 6309.57 nM T41580 CO9VA3 9820671 IC50 > 1000 nM T41580 C6KJ7P 9827677 Ki = 145 nM T41580 CQZ6I0 9828476 Ki = 218.78 nM T41580 CS3MA5 9837106 Ki = 940 nM T41580 CB7L9H 9846548 Ki = 42 nM T41580 CY2D5T 9851486 Ki = 436.52 nM T41580 CV2HW7 9883506 Ki = 18 nM T41580 CTAC24 9885114 Ki = 368 nM T41580 C8HS4Q 9895326 Ki = 257.04 nM T41580 CYWQ50 9906447 Ki > 10000 nM T41580 C7JFZ5 9906978 Ki = 1543 nM T41580 C7SMT0 9908904 IC50 > 1000 nM T41580 C32ZXG 9923679 Ki = 3700 nM T41580 C03ZFH 9931977 Ki = 376 nM T41580 CUQ8I5 9947861 Ki < 6309.57 nM T41580 CO2X8D 9951544 IC50 = 11.48 nM T41580 CF1C5Q 9960497 Ki = 570 nM T41580 C3O9SC 9971924 Ki = 141.25 nM T41580 C2EUY0 10035109 Ki > 10000 nM T41580 C5MZ6I 10042547 Ki = 4168.69 nM T41580 C7D0GO 10044968 Ki = 1280 nM T41580 CB82XU 10045088 Ki > 10000 nM T41580 C3MTF4 10045713 Ki = 1330 nM T41580 CLE0M4 10056237 Ki = 18.6 nM T41580 CZ0U2N 10070896 Ki = 1700 nM T41580 C7J1UB 10101373 Ki = 990 nM T41580 COF5U3 10109188 Ki > 10000 nM T41580 C3N8JR 10123375 Ki = 166.2 nM T41580 C9XCB3 10132386 Ki > 5000 nM T41580 CE27RV 10135864 EC50 > 10000 nM T41580 CNB56M 10177445 Ki = 3900 nM T41580 C7MKP9 10199335 Ki < 6309.57 nM T41580 CLY2B9 10220232 Ki = 100 nM T41580 CU2B9P 10221004 Ki < 6309.57 nM T41580 CX9YD5 10221005 Ki < 6309.57 nM T41580 C0LOA6 10251036 Ki = 420 nM T41580 C6G0AY 10266032 Ki = 32.36 nM T41580 CBE9K1 10317643 Ki > 10000 nM T41580 C4MD0S 10318507 Ki = 880 nM T41580 CSU1R6 10319299 Ki > 10000 nM T41580 C6W5DM 10333157 Ki = 588.84 nM T41580 C3E5CB 10337773 Ki = 25118.86 nM T41580 C1A3KN 10350094 Ki = 134.3 nM T41580 COS13I 10362866 Ki = 580 nM T41580 C4H6YF 10379435 Ki < 6309.57 nM T41580 C3N7TF 10382537 Ki = 42.66 nM T41580 CIQ02H 10436842 Ki = 288 nM T41580 CIDE58 10473701 Ki = 1270 nM T41580 C8FA2T 10474679 Ki = 1900 nM T41580 CBS8U6 10475736 Ki = 1750 nM T41580 CJ0K1T 10507651 Ki = 380.19 nM T41580 C2U8AC 10508016 Ki = 891.25 nM T41580 C4XZ3Y 10508132 Ki = 1819.7 nM T41580 CZP09X 10508332 Ki = 575.44 nM T41580 C4X9EF 10531532 Ki = 512.86 nM T41580 C7MI2N 10531766 Ki = 870.96 nM T41580 CF24MW 10579368 Ki = 199.53 nM T41580 CK8SO7 10603951 Ki = 489.78 nM T41580 CB26QH 10626982 Ki = 831.76 nM T41580 CSWC40 10627021 Ki = 912.01 nM T41580 CF1P6Z 10651080 Ki = 204.17 nM T41580 C3K7UP 10651654 Ki = 1258.93 nM T41580 CTB7L2 10674896 Ki = 1258.93 nM T41580 C3IX8A 10707358 Ki = 6.918 nM T41580 CT1K3B 10769331 Ki = 91.2 nM T41580 C3O7YN 10793665 Ki = 2290.87 nM T41580 C0D6MW 10793963 Ki = 371.54 nM T41580 CBO8N9 10818003 Ki = 380.19 nM T41580 CE80NV 10841190 Ki = 1513.56 nM T41580 CYSL64 10841387 Ki = 912 nM T41580 C5AY9R 10848826 Ki = 40.74 nM T41580 C8VT6G 10916464 Ki < 6309.57 nM T41580 CH95TI 10923927 Ki < 6309.57 nM T41580 C3CI6Z 10934575 Ki = 977.24 nM T41580 CGW87Y 11034737 Ki = 1659.59 nM T41580 CA7IB5 11043720 Ki = 1258.93 nM T41580 C48QYR 11058166 Ki < 6309.57 nM T41580 C7JI1M 11059195 Ki < 6309.57 nM T41580 C7R2AZ 11079593 Ki < 6309.57 nM T41580 C91BKL 11090351 Ki < 6309.57 nM T41580 CFE1M7 11097789 Ki = 851.14 nM T41580 CTG4I5 11098175 Ki < 6309.57 nM T41580 CR6K4V 11109088 Ki = 676.08 nM T41580 C6SXJ0 11140033 Ki = 1148.15 nM T41580 CG40BP 11140345 Ki = 3981.07 nM T41580 CO0XW1 11140347 Ki = 331.13 nM T41580 CTA5J4 11173544 Ki = 398.11 nM T41580 CU86DN 11173568 Ki = 478.63 nM T41580 C5JYO7 11186227 Ki = 812.83 nM T41580 C3ALW8 11199581 Ki = 1000 nM T41580 C9T7YZ 11199593 Ki = 3548.13 nM T41580 C5YQ0F 11203101 Ki = 1300 nM T41580 C62KQF 11211035 Ki = 269.15 nM T41580 CEGZ35 11221758 Ki = 1548.82 nM T41580 C59VOU 11225732 Ki = 949 nM T41580 COCU26 11246610 Ki = 501.19 nM T41580 CNTE30 11265631 Ki = 933.25 nM T41580 C8SYW5 11277479 Ki = 537.03 nM T41580 C84NSM 11278634 Ki < 10000 nM T41580 CNAQ56 11293787 Ki = 299 nM T41580 CA1D3O 11300487 Ki = 831.76 nM T41580 C3JBI0 11338418 Ki > 500 nM T41580 C96OKG 11346584 Ki = 354.81 nM T41580 CV17WA 11360447 Ki = 213.8 nM T41580 CI69GW 11361608 Ki = 660.69 nM T41580 CA28SQ 11371902 Ki = 416.87 nM T41580 C9U5WT 11380132 Ki = 3311.31 nM T41580 C1ZOY6 11380133 Ki = 2691.53 nM T41580 CB01AS 11448533 Ki = 10000 nM T41580 CX8CN6 11473729 Ki = 10000 nM T41580 CZA0M9 11653915 Ki = 7.3 nM T41580 CJ1KW9 11741010 Ki = 910 nM T41580 CPG15O 11743399 IC50 > 1000 nM T41580 CIM1E0 11750482 Ki = 160 nM T41580 CJ58LT 11765813 Ki = 46 nM T41580 CFTI34 11801828 Ki = 575.44 nM T41580 C1VWL5 11811395 Ki < 6309.57 nM T41580 C8JQL7 11957735 IC50 > 10000 nM T41580 CGY20U 12114850 Ki = 1510 nM T41580 CNS58C 12114851 Ki = 188.6 nM T41580 CVY50Z 12114852 Ki = 27.6 nM T41580 C7DQR1 12114853 Ki = 44.7 nM T41580 CIUR20 12699315 Ki = 1318.26 nM T41580 C2V9FL 13091268 Ki = 515.5 nM T41580 CWBX46 13123534 EC50 = 776.25 nM T41580 C1CX2S 15675860 Ki = 323.59 nM T41580 CXM74T 16090594 Ki = 1320 nM T41580 C8QLC1 16090595 Ki = 1150 nM T41580 C01RFM 16090596 Ki = 1100 nM T41580 CAYX52 16090597 Ki = 3600 nM T41580 CW0U8R 16090598 Ki = 1120 nM T41580 C06KXJ 16090599 Ki = 2500 nM T41580 COB96N 16090600 Ki = 1680 nM T41580 C6YPM3 16090601 Ki = 1800 nM T41580 CR02MW 16090602 Ki = 2600 nM T41580 CC5HV2 16090621 Ki = 96 nM T41580 COTF82 16090622 Ki = 3500 nM T41580 CB2Z6H 16090623 Ki = 600 nM T41580 C4WAZ1 16090624 Ki = 2600 nM T41580 C6MH3Z 16090625 Ki = 2030 nM T41580 CX98OC 16090626 Ki = 3470 nM T41580 C6D0WK 16090627 Ki = 2900 nM T41580 C1B5TL 16090628 Ki = 2600 nM T41580 CTXU32 16090630 Ki = 1470 nM T41580 CD8FX2 16090631 Ki = 5100 nM T41580 C63QEJ 16090632 Ki = 17600 nM T41580 C98XNF 16090633 Ki = 3150 nM T41580 C1G7KL 16090634 Ki > 30000 nM T41580 C8YBI4 16090635 Ki = 2980 nM T41580 CZ2IS9 16660294 Ki > 10000 nM T41580 CVU96E 16725934 Ki = 752 nM T41580 CFMX86 16757089 Ki = 741.31 nM T41580 C6OJ3A 16757182 Ki = 1584.89 nM T41580 CPRJ25 21392988 Ki = 11748.98 nM T41580 C3T5HF 21509921 Ki = 413 nM T41580 CT7XG9 21830793 Ki = 238 nM T41580 C8GUJ3 22120322 IC50 = 1.549 nM T41580 CGO3B8 22120332 IC50 = 2.042 nM T41580 C02AEX 22493245 Ki < 6309.57 nM T41580 CF9D1U 23622576 Ki = 190.55 nM T41580 CDC91N 24839550 Ki = 302 nM T41580 CY21RE 24841480 Ki = 800 nM T41580 C2C7WN 24882007 Ki = 79 nM T41580 C8WH5Z 24906160 Ki = 1202.26 nM T41580 C3RQ1P 24906196 Ki = 446.68 nM T41580 CBT65R 24906197 Ki = 870.96 nM T41580 C9OAG1 24906198 Ki = 338.84 nM T41580 CYL83G 24906199 Ki = 190.55 nM T41580 CC9W0R 24906200 Ki = 954.99 nM T41580 CYEA86 24906201 Ki = 1071.52 nM T41580 CIR8G1 24906202 Ki = 1659.59 nM T41580 CPH75D 24906203 Ki = 1000 nM T41580 CBUH25 24906241 Ki = 478.63 nM T41580 CUNP93 24906242 EC50 = 15848.93 nM T41580 C7Y2SB 24906243 Ki = 1071.52 nM T41580 C1VRJ3 25014630 IC50 = 32000 nM T41580 C9XMH7 25110718 Ki = 14.3 nM T41580 CX04LB 25142456 Ki = 10 nM T41580 CWT9F7 28918670 Ki = 616.6 nM T41580 CAM63X 42618195 IC50 > 1000 nM T41580 C8K4UF 42618197 IC50 > 1000 nM T41580 CW4ST6 42636938 EC50 = 4200 nM T41580 CJ3NP5 42636941 IC50 = 954.99 nM T41580 C2AV1K 44190762 IC50 = 770 nM T41580 C9O1RI 44215744 Ki = 49 nM T41580 CK7F2E 44240743 IC50 = 7500 nM T41580 CO65VL 44269006 Ki = 707.95 nM T41580 C0TP2Z 44269013 Ki = 549.54 nM T41580 CW6A9E 44269089 EC50 = 251.19 nM T41580 CZ63DE 44269122 Ki = 165.96 nM T41580 CDS8G5 44269140 Ki = 1584.89 nM T41580 CZ5P6U 44288769 Ki = 955 nM T41580 CZ7O4D 44288847 Ki = 676 nM T41580 C6DYQ1 44288874 Ki = 531 nM T41580 CAG7E1 44288877 Ki = 1758 nM T41580 CQ3Y5R 44288945 Ki = 162 nM T41580 C5ZL4A 44289035 Ki = 776 nM T41580 CLRZ30 44292232 Ki = 91.2 nM T41580 C7GUL1 44292381 Ki = 22.39 nM T41580 C3G1KO 44292385 Ki = 40.74 nM T41580 C0R8WU 44292386 Ki = 102.33 nM T41580 C6G8ZC 44311789 Ki = 18197.01 nM T41580 C5L1WN 44312036 Ki = 3235.94 nM T41580 CT46CK 44312037 Ki = 17378.01 nM T41580 C3XFH4 44312198 Ki = 85113.8 nM T41580 CZ4TN0 44314198 Ki = 5.888 nM T41580 CCI07K 44314200 Ki = 25.12 nM T41580 CA56FM 44324725 Ki = 42 nM T41580 CW16JD 44324737 Ki = 14 nM T41580 CA84SN 44324765 Ki = 14 nM T41580 COA3H4 44324800 Ki = 3 nM T41580 CK32IL 44324859 Ki = 315 nM T41580 CMB1S6 44324860 Ki > 1000 nM T41580 C8HUD2 44324887 Ki = 12 nM T41580 CCT53K 44324900 Ki = 995 nM T41580 CL1F3T 44324906 Ki = 16 nM T41580 CPAL75 44324937 Ki = 2 nM T41580 CY04JW 44324972 Ki = 14 nM T41580 C76UJT 44325027 Ki > 1000 nM T41580 C1RS8C 44325028 Ki > 1000 nM T41580 CR4Q1C 44325038 Ki = 721 nM T41580 C4SZJ2 44325044 Ki = 370 nM T41580 CQX1Y0 44325049 Ki = 31 nM T41580 C0N3JG 44325050 Ki = 7.5 nM T41580 CGS4E7 44325079 Ki > 1000 nM T41580 CZ2X3A 44352155 EC50 = 954.99 nM T41580 C67ZNM 44352207 Ki = 501.19 nM T41580 C6KJV8 44371744 Ki = 275.42 nM T41580 CI90WF 44371745 Ki = 281.84 nM T41580 C09ADW 44371755 Ki = 181.97 nM T41580 CUF64I 44371848 Ki = 18.5 nM T41580 C76VTG 44371864 Ki = 269.15 nM T41580 C3K6GE 44376845 IC50 = 194.98 nM T41580 CPD18R 44376900 IC50 = 1.738 nM T41580 CE46SW 44376923 IC50 = 1.479 nM T41580 C7UW8Z 44376927 IC50 = 1.95 nM T41580 C8GT5O 44376936 IC50 = 10.72 nM T41580 CLC2T4 44376954 IC50 = 2.63 nM T41580 C9IPC3 44376958 IC50 = 2.57 nM T41580 CX4A1Z 44376975 IC50 = 4.169 nM T41580 C14SMK 44376984 IC50 = 2.089 nM T41580 C0V4XL 44376993 IC50 = 1.259 nM T41580 CX0UR3 44377006 IC50 = 79.43 nM T41580 CB2R0M 44377007 IC50 = 4.365 nM T41580 C2ID6U 44377035 IC50 = 2.138 nM T41580 C6R9OZ 44377036 IC50 = 0.955 nM T41580 C97QIG 44377200 IC50 = 1.349 nM T41580 CI47TG 44421258 Ki = 19952.62 nM T41580 CK7HF3 44424855 Ki = 14 nM T41580 C28OZL 44438147 Ki = 370 nM T41580 CKB9O7 44438148 Ki = 330 nM T41580 C1AR8P 44438152 Ki = 804 nM T41580 CZR64Y 44438161 Ki = 584 nM T41580 CG38YN 44438165 Ki = 2068 nM T41580 C8RC7O 44438166 Ki = 1535 nM T41580 C5GPZ7 44438167 Ki = 857 nM T41580 C0QI8L 44438168 Ki = 1364 nM T41580 C12XGE 44456400 Ki = 243 nM T41580 C4LUK7 44549156 Ki = 309.03 nM T41580 C8N3ID 44568614 Ki = 47.86 nM T41580 CWM4U7 44579184 Ki = 17 nM T41580 CLO8A9 44579185 Ki = 49 nM T41580 CGVM03 44579186 Ki = 8 nM T41580 CM6L2Y 44579187 Ki = 27.5 nM T41580 CBDL39 44579228 Ki = 28 nM T41580 CX5O1H 44579229 Ki = 10.5 nM T41580 C3G5YK 44579230 Ki = 10.9 nM T41580 CKTJ23 44579231 Ki = 17.9 nM T41580 C57BWM 44579271 Ki = 69.5 nM T41580 C7R9XM 44579272 Ki = 5.2 nM T41580 CWO70X 45260703 Ki < 6309.57 nM T41580 C4VOW6 45260704 Ki = 2344.23 nM T41580 CQ0R5Y 45264581 Ki = 776.25 nM T41580 C39CDN 45264638 Ki = 1621.81 nM T41580 CQHW85 45487089 Ki = 269.15 nM T41580 CI34PT 45487144 Ki = 165.96 nM T41580 CC9GH0 45487145 Ki = 338.84 nM T41580 C7MZ9Y 45487955 Ki = 537.03 nM T41580 CLW5M9 45487956 Ki = 309.03 nM T41580 C45DAV 45487958 Ki = 398.11 nM T41580 CZSW97 45487962 EC50 = 61.66 nM T41580 C03LTM 46869265 Ki = 6400 nM T41580 C8VUO2 49781004 Ki = 23.99 nM T41580 C0LAT9 49781005 Ki = 2.818 nM T41580 C12UVE 49781006 Ki = 9.772 nM T41580 CW1V4K 49781007 Ki = 6.457 nM T41580 CF9L7Z 49781008 Ki = 11.75 nM T41580 CQ2EN5 49781222 Ki = 0.6918 nM T41580 CV62OU 49781223 Ki = 1.622 nM T41580 C3I5HP 49781224 Ki = 2.291 nM T41580 CF5CO4 49781228 Ki = 0.1096 nM T41580 CW5X6A 49781887 Ki = 1.905 nM T41580 C2LZJ0 49783209 Ki = 671.2 nM T41580 C57SMG 49783415 Ki > 10000 nM T41580 C0TG6I 49783419 Ki = 773 nM T41580 C28CKM 49836301 Ki = 398.11 nM T41580 C5JO6E 49836302 Ki = 562.34 nM T41580 C9TNO4 49836303 Ki = 263.03 nM T41580 CL6QA1 49836304 Ki = 562.34 nM T41580 CE1S9B 49836305 Ki = 446.68 nM T41580 CP0DJ4 49836306 Ki = 707.95 nM T41580 CJM3F9 49836307 Ki = 1000 nM T41580 C0LN3I 49836308 Ki = 316.23 nM T41580 C2RY0J 50878551 Ki = 724.44 nM T41580 C1W6TV 50898777 Ki = 1258.93 nM T41580 CXMZ73 50898778 Ki > 10000 nM T41580 CE4KP1 51050257 Ki > 10000 nM T41580 CR8MI3 52941512 Ki = 0.2042 nM T41580 CZ4SA1 52942940 Ki = 1230.27 nM T41580 CH3YE5 52943739 Ki = 0.912 nM T41580 C70LBS 52944548 Ki = 0.182 nM T41580 C7WN4S 52948958 Ki = 0.3467 nM T41580 C5W7SH 52950140 Ki = 1.148 nM T41580 C6PUX9 56645570 IC50 = 2490 nM T41580 C2KG9D 56665110 Ki > 10000 nM T41580 C1TC7Q 56963799 Ki > 10000 nM T41580 C4RBY6 57345625 EC50 = 162.18 nM T41580 C1US6F 57345626 EC50 = 316.23 nM T41580 CNU83J 57345627 Ki = 870.96 nM T41580 CD50GK 57345628 Ki = 407.38 nM T41580 C4FA1T 57345629 Ki = 1047.13 nM T41580 CO2W7Z 57384051 Ki > 10000 nM T41580 C80DHR 57393066 Ki > 10000 nM T41580 C4N0TW 57393922 EC50 = 3162.28 nM T41580 C6X0ZI 57394788 Ki > 10000 nM T41580 CR6U3P 57394789 Ki > 10000 nM T41580 CH84EC 57395663 EC50 = 239.88 nM T41580 CL37YV 57395731 EC50 = 295.12 nM T41580 C5I3DG 57395732 EC50 = 199.53 nM T41580 CR1Y7M 57398332 Ki > 10000 nM T41580 CM9WK5 57399145 Ki = 1318.26 nM T41580 CIB2L3 57399991 Ki > 10000 nM T41580 CQ7MC1 57400959 EC50 = 10000 nM T41580 C9WE2A 57401787 Ki = 4466.84 nM T41580 C56WAY 57402717 Ki = 870.96 nM T41580 C1BFP4 57402718 EC50 = 316.23 nM T41580 CP21KC 57403508 Ki = 2818.38 nM T41580 C2PJ4N 59271992 IC50 = 1000 nM T41580 C3XL7O 66561967 Ki = 4241 nM T41580 CLM79R 70686398 Ki > 10000 nM T41580 CJQX48 70693375 Ki = 338.84 nM T41580 CST13M 70695474 Ki = 407.38 nM T41580 C6CNI0 70696790 Ki = 2818.38 nM T41580 C5L8NJ 72947314 Ki = 501.19 nM T41580 CE1JY2 72947315 Ki = 794.33 nM T41580 CC65OA 73213195 Ki = 2187 nM T41580 CW83DK 73213196 Ki = 4354 nM T41580 C02FTM 73291731 Ki = 537.03 nM T41580 CCV91B 73346042 Ki = 56.2 nM T41580 CVKN29 73346335 Ki > 10000 nM T41580 CW8A0Y 73349359 Ki = 665 nM T41580 C6BS5L 73349361 Ki = 1274 nM T41580 CV1U7L 73352414 Ki = 2535 nM T41580 C1NJ0R 73353884 Ki = 3256 nM T41580 C4F7VK 73355415 Ki = 1005 nM T41580 C8IDL3 75306277 Ki = 199.53 nM T41580 CUQ6V0 92042918 Ki < 1000 nM T41580 C7YQM3 101333429 Ki = 1230 nM T41580 CWR6I1 118112300 IC50 = 8000 nM T41580 CCY5S0 118717248 Ki = 72 nM T41580 CCR09Q 118717249 Ki = 158 nM T41580 C5X8MN 122186880 Ki = 3220 nM T41580 C7ODW3 122195524 Ki > 900 nM T41580 CM57GR 126720252 Ki = 984 nM T41580 CTBN56 127026052 Ki = 218.78 nM T41580 C8MC1I 127028408 Ki = 380.19 nM T41580 CQ0ZT9 127035062 Ki = 29 nM T41580 CU49VE 127036186 Ki = 436.52 nM T41580 CG06BD 127036932 Ki = 169.82 nM T41580 CVW71O 127036953 Ki = 229.09 nM T41580 C4RV9T 129928082 EC50 = 3162.28 nM T41580 C1RI8Q 132060720 Ki = 1444 nM T41580 C0DIF5 132060733 Ki = 3343 nM T41580 CY8B9L 132060743 Ki = 454 nM T41580 C7FM0U 132060763 Ki = 2439 nM T41580 CT81OY 132060776 Ki = 2285 nM T41580 CFXL21 132060812 Ki > 10000 nM T41580 C7CSU4 132075278 Ki = 2985 nM T41580 CAVB41 132584404 Ki = 1040 nM T41580 CS3FI6 134137108 EC50 = 4570.88 nM T41580 CBU81N 134149168 Ki > 10000 nM T41580 CFG4Y1 134156190 EC50 = 2511.89 nM T41580 CP58JO 135418497 Ki = 116 nM T41580 C9H8ZO 135423051 Ki = 9300 nM T41580 CH96LU 135559170 Ki = 253 nM T41580 C5J9BC 136019934 Ki = 4.5 nM T41580 CE8N4S 137641762 Ki = 5000 nM T41580 CPI68E 137646281 Ki = 241 nM T41580 CR9F3Q 137653203 Ki = 5000 nM T41580 C4GV8Q 145990586 Ki = 571 nM T41580 C6P3SR 153287553 Ki > 10000 nM T41580 CV9G7Z 153287572 Ki > 10000 nM T41580 CO85KL 153287574 Ki = 398.11 nM T41580 CUSA24 155519891 Ki > 10000 nM T41580 CB79ZW 155536080 Ki = 5011.87 nM T41580 CA8JO5 155540582 IC50 = 790 nM T41580 CZ49CM 155545843 Ki = 1720 nM T41580 CP9TR0 10324985 Ki = 316.2 nM T41580 D00GEE 92766 Ki = 455 nM T41580 D01KAX 135453290 EC50 = 3050 nM T41580 D03DMN 1268096 Ki = 116 nM T41580 D03LDH 10758200 Ki = 72.8 nM T41580 D05GDP 599482 Ki = 140 nM T41580 D05ZUX 44207909 Ki >= 1000 nM T41580 D06QKW 2765 Ki = 524.81 nM T41580 D06UBB 123981 Ki = 16 nM T41580 D07ICV 3072540 Ki = 1200 nM T41580 D07QCC 10946567 Ki = 15 nM T41580 D08KLH 108094 Ki = 1.622 nM T41580 D09RPR 16737207 Ki > 10000 nM T41580 D0D8GV 9830741 Ki > 45 nM T41580 D0E3OL 4567175 Ki = 3800 nM T41580 D0FF6S 16038374 IC50 > 10000 nM T41580 D0FU5E 10220053 Ki = 23 nM T41580 D0H3CW 9839317 Ki = 14 nM T41580 D0H3NA 10176567 Ki = 663 nM T41580 D0L5MW 181743 Ki = 252 nM T41580 D0L7IZ 540335 Ki = 1500 nM T41580 D0LI3J 3080926 Ki = 26915.35 nM T41580 D0M5ZE 5311416 Ki = 2511.89 nM T41580 D0N7UE 10198248 Ki = 218.78 nM T41580 D0PN9R 16655023 Ki = 1.5 nM T41580 D0T2RY 9948320 Ki = 840 nM T41580 D0V6DJ 5640 Ki = 406 nM T41580 D0Y0SA 135399666 EC50 = 4710 nM T41580 D0Z7EA 643606 Ki = 4.7 nM T20331 D02NMO 10421577 IC50 = 427 nM T20331 D0I5HE 9884833 IC50 = 3 nM T20331 D0K4NZ 20629114 Ki = 5 nM T20331 D0V2GT 5311023 Ki > 10000 nM T20331 CT6RA0 2317 Ki = 5000 nM T20331 C9NG4X 16033 EC50 = 3.162 nM T20331 C8GL7K 213847 IC50 = 80 nM T20331 CFBM96 296732 Ki = 34 nM T20331 C74KDN 624746 Ki = 33 nM T20331 CO6FY2 794166 IC50 > 1000 nM T20331 C1U0HV 1284592 IC50 = 1600 nM T20331 C1Q4WZ 1294837 Ki > 5011.87 nM T20331 CYT2I0 1639804 IC50 = 7 nM T20331 CEP31Y 2226619 Ki = 14 nM T20331 CK49PQ 2821670 IC50 = 59 nM T20331 C3EGK1 3087469 IC50 = 100 nM T20331 CF20QJ 4527770 Ki = 15.85 nM T20331 C39UDN 5312114 IC50 = 1.3 nM T20331 CD0LO7 9796081 IC50 = 1.1 nM T20331 C6TE5S 9796164 IC50 = 1.7 nM T20331 CI26VT 9799669 IC50 = 69 nM T20331 CPCH23 9801629 IC50 = 8.8 nM T20331 CA1VW4 9802118 IC50 = 1.5 nM T20331 C5MC8Y 9802119 IC50 = 1.5 nM T20331 C4HSU8 9805850 IC50 = 37 nM T20331 CJ2KX8 9806472 Ki = 14 nM T20331 C4GHT3 9806525 IC50 = 36 nM T20331 CYBG93 9806557 IC50 = 236 nM T20331 C1NQC6 9807658 IC50 = 2400 nM T20331 CX02ZK 9810707 IC50 = 11 nM T20331 CNLU01 9819988 IC50 = 9300 nM T20331 CAX4E3 9821993 Ki = 7.4 nM T20331 C0PL9I 9822252 IC50 = 3.7 nM T20331 CU8BQ5 9823032 IC50 = 1.7 nM T20331 CHI0O9 9824246 IC50 = 15 nM T20331 CS4DX3 9825755 IC50 = 60 nM T20331 CAT86W 9825886 IC50 = 2.4 nM T20331 CKMH19 9827743 IC50 = 6 nM T20331 C2YPQ8 9845943 Ki = 1.1 nM T20331 CH84YW 9847327 Ki = 7.5 nM T20331 C5LQA7 9847333 IC50 = 9 nM T20331 CC9D4R 9850107 IC50 = 10 nM T20331 CECS52 9857217 IC50 = 13 nM T20331 C20JKX 9858246 Ki = 15 nM T20331 CKAZ42 9862646 IC50 = 2 nM T20331 CIO9N8 9866472 IC50 = 5.7 nM T20331 CK7QY8 9867212 IC50 = 5 nM T20331 CV17EX 9868487 IC50 = 0.47 nM T20331 CT7S5I 9869041 IC50 > 10000 nM T20331 C7C6OL 9869232 IC50 = 0.85 nM T20331 CA5E4O 9871208 IC50 = 52 nM T20331 C6DQR2 9871512 IC50 = 75 nM T20331 CY7WL0 9880835 IC50 = 7.2 nM T20331 CA86RB 9880873 IC50 = 560 nM T20331 C0XYG6 9882119 IC50 = 0.7 nM T20331 CXJL03 9885994 IC50 = 6.5 nM T20331 C5DG2E 9886573 IC50 = 1.9 nM T20331 CPGD84 9887225 Ki = 2.4 nM T20331 C2SPB9 9887226 IC50 = 4.2 nM T20331 CCZ60M 9887852 Ki = 0.9 nM T20331 CU1I6O 9888553 Ki = 1.1 nM T20331 C2J8AU 9888989 IC50 ~ 1000 nM T20331 CD7M3B 9889156 IC50 = 0.91 nM T20331 CD26ME 9890550 IC50 = 4.1 nM T20331 C5HJ3U 9891987 IC50 = 22 nM T20331 CZ3RF9 9892202 IC50 = 28 nM T20331 CY1P7H 9895868 IC50 = 2.7 nM T20331 C0XWF1 9902517 IC50 = 54 nM T20331 C57AHB 9903829 IC50 = 36 nM T20331 C2W9FL 9905079 IC50 = 52 nM T20331 CPA61I 9907999 Ki = 3.5 nM T20331 CU83VQ 9908374 IC50 = 0.84 nM T20331 C27WHT 9908720 IC50 = 80 nM T20331 C3RE1D 9908801 IC50 = 0.9 nM T20331 CYC62U 9908890 IC50 = 1.5 nM T20331 C8KYH2 9908945 IC50 = 1.4 nM T20331 C03YEQ 9908946 IC50 = 2 nM T20331 CS92LR 9916525 Ki > 10000 nM T20331 CJ67UW 9922092 Ki = 93 nM T20331 CW84OK 9922187 Ki = 21 nM T20331 CIW81R 9923839 IC50 = 2.4 nM T20331 C1QB7U 9924211 IC50 = 19 nM T20331 CQ13GT 9924627 IC50 = 10 nM T20331 CF2M1T 9926566 IC50 = 1.8 nM T20331 CWP3V6 9930778 Ki = 1.2 nM T20331 CN0B7S 9930807 IC50 = 0.64 nM T20331 C52LMX 9930851 IC50 = 2.1 nM T20331 CZMP76 9933356 IC50 = 1.8 nM T20331 C4L1GA 9934033 IC50 = 2700 nM T20331 C8CUH6 9934437 IC50 = 21 nM T20331 CAY3G0 9934923 IC50 = 9 nM T20331 C5E8OF 9936263 IC50 = 25 nM T20331 CZ4X5D 9946965 IC50 = 2 nM T20331 CJ9V1G 9947073 IC50 = 8.7 nM T20331 CT76GZ 9947469 IC50 = 5.4 nM T20331 C39RLP 9949840 IC50 = 220 nM T20331 C9WRJ1 9952193 Ki = 8.3 nM T20331 C5C2PJ 9952231 IC50 = 4.4 nM T20331 CP5X6F 9952232 IC50 = 1.3 nM T20331 CIT45Q 9952815 IC50 = 1.8 nM T20331 C02XWA 9953150 IC50 = 1.2 nM T20331 CFH0D1 9953800 IC50 = 1.1 nM T20331 C4O6FD 9953802 IC50 = 1.8 nM T20331 CJ8N4V 9955287 IC50 = 1.9 nM T20331 C06PRD 9955360 IC50 = 28 nM T20331 C7HOD0 9957190 IC50 = 0.68 nM T20331 CUSA49 9967563 IC50 = 47 nM T20331 C6SU4K 9967784 IC50 = 93 nM T20331 CU35AC 9969726 IC50 = 69 nM T20331 CGLQ63 9972871 Ki = 8 nM T20331 CX3JC1 9979057 IC50 = 1.7 nM T20331 CC05RX 9982218 Ki = 8 nM T20331 C72HXY 10005032 Ki = 32 nM T20331 CH1Q6E 10008757 Ki > 10000 nM T20331 C54LEF 10017062 Ki = 10 nM T20331 CM6U4F 10020909 Ki = 101 nM T20331 CK3W5X 10030299 Ki > 10000 nM T20331 C7BL3Z 10040233 IC50 = 0.5 nM T20331 CHUI86 10041217 Ki = 1.5 nM T20331 C05SFO 10041884 Ki = 41 nM T20331 CTON52 10045322 Ki = 13 nM T20331 C04HZE 10046270 Ki = 2.8 nM T20331 CZ4SN6 10047390 IC50 = 150 nM T20331 C73QBA 10047509 Ki = 2.8 nM T20331 CUFC30 10051692 IC50 = 7.7 nM T20331 C7VHZ4 10062681 Ki = 1.6 nM T20331 C82VAF 10071200 IC50 = 12.5 nM T20331 CL96TH 10110741 IC50 = 6400 nM T20331 C47JRT 10111188 Ki = 52 nM T20331 C04RFK 10111791 IC50 = 4 nM T20331 CNCK67 10111792 IC50 = 2 nM T20331 C52EPR 10111849 IC50 = 25 nM T20331 CR1AI7 10112368 Ki = 35 nM T20331 C9ZU5Q 10112931 Ki = 2 nM T20331 C1EHM4 10133076 IC50 = 2.7 nM T20331 C2W7AM 10139215 IC50 = 4 nM T20331 CI6S1O 10139329 Ki = 3.2 nM T20331 CMI3U1 10154767 IC50 = 30 nM T20331 CFG9Y2 10155282 Ki = 2.6 nM T20331 C21SKI 10155286 Ki = 59 nM T20331 C8K1VL 10159053 IC50 = 28 nM T20331 CC3F4X 10159722 Ki = 1.2 nM T20331 C85KSE 10160875 Ki = 160 nM T20331 C73ZCO 10161574 Ki = 3.4 nM T20331 CT42AQ 10161870 IC50 = 30 nM T20331 CW0OK6 10178465 Ki = 3 nM T20331 CY2K6R 10181110 Ki = 3.2 nM T20331 C9LBU7 10183204 Ki = 48 nM T20331 C9C5JX 10186456 IC50 = 10 nM T20331 CQ92PA 10202456 Ki = 2.6 nM T20331 C9V3TM 10202875 Ki = 13 nM T20331 CMY83E 10203845 Ki = 0.75 nM T20331 C7PB9K 10205608 Ki = 8.8 nM T20331 CC9VQ7 10223183 Ki = 20 nM T20331 CH6RC1 10223395 IC50 = 9.2 nM T20331 C5NAL0 10223847 Ki = 27 nM T20331 CG2WN7 10224063 Ki = 5.9 nM T20331 CAN6X3 10226374 IC50 = 2 nM T20331 CNHR93 10231050 IC50 > 1000 nM T20331 CEI7C4 10245014 Ki = 15 nM T20331 CTE92X 10247746 Ki = 12 nM T20331 CR0HX4 10255890 IC50 = 0.23 nM T20331 C9H3XN 10266238 IC50 = 0.4 nM T20331 C4EJH5 10272418 IC50 = 2 nM T20331 C0CKW7 10272799 Ki = 1.5 nM T20331 C2B4JF 10273149 IC50 = 4.8 nM T20331 CT1IA8 10273848 Ki = 0.4 nM T20331 CU9NY6 10275303 Ki = 2.8 nM T20331 C87WIR 10293081 IC50 = 4.3 nM T20331 C6IXU4 10293988 Ki = 1.8 nM T20331 C1JR3H 10294504 IC50 = 6.2 nM T20331 COU3E8 10294889 Ki = 6.3 nM T20331 C8L7WY 10295464 IC50 = 7 nM T20331 CDJE64 10295943 Ki = 311 nM T20331 C3J7EG 10298415 Ki = 1.1 nM T20331 CFJ98P 10298981 IC50 = 24 nM T20331 C3ZJY6 10303307 IC50 = 1800 nM T20331 CUD3N9 10332613 Ki = 16 nM T20331 CGZT74 10336953 Ki = 43 nM T20331 C4IPC0 10341402 Ki = 6.6 nM T20331 C86KRU 10363209 Ki = 2.9 nM T20331 CX34PS 10364093 Ki = 4.7 nM T20331 CZM0K4 10384590 Ki = 16 nM T20331 CA1C6E 10418848 Ki > 1000 nM T20331 C4HMY5 10429613 IC50 = 45 nM T20331 CAXE13 10430847 IC50 = 232 nM T20331 CZQ45W 10432823 Ki = 8.5 nM T20331 C2ZHJ3 10435289 Ki = 12 nM T20331 CRNL80 10449735 Ki = 38 nM T20331 C8R1IL 10450609 Ki = 15 nM T20331 CRF1A2 10451123 IC50 = 218 nM T20331 CNR16C 10457755 IC50 = 11.5 nM T20331 C0Q1JD 10471957 IC50 = 0.3 nM T20331 CZ85WP 10477251 IC50 = 2.6 nM T20331 CIF3E6 10496226 IC50 = 4700 nM T20331 CMY5O1 10497816 IC50 = 44 nM T20331 CX6RE7 10498512 IC50 = 28 nM T20331 CGD4L2 10498514 IC50 = 8300 nM T20331 C37JDR 10498644 IC50 = 18 nM T20331 C6LD4N 10500401 IC50 = 7800 nM T20331 C0A2GD 10517831 IC50 = 470 nM T20331 CMC18P 10518886 IC50 = 540 nM T20331 C4EZ1S 10519375 IC50 = 2300 nM T20331 COW2X7 10519637 IC50 = 1100 nM T20331 C31UYP 10520484 IC50 = 1400 nM T20331 CER48F 10522130 IC50 = 32 nM T20331 C8P2KB 10522285 IC50 = 330 nM T20331 CGV51K 10522705 IC50 < 0.1 nM T20331 C84MSG 10524003 Ki > 10000 nM T20331 CKQ2G1 10531484 Ki > 10000 nM T20331 C6IFC1 10547234 IC50 = 120 nM T20331 CU25ZB 10549405 IC50 = 7500 nM T20331 CQ1P5I 10554658 Ki > 10000 nM T20331 C0F9SD 10555187 Ki > 10000 nM T20331 C1TRN7 10565529 IC50 = 1.7 nM T20331 CJD36Q 10571295 IC50 = 6000 nM T20331 CB1E2N 10572176 IC50 = 5200 nM T20331 CD59XU 10573317 IC50 = 1400 nM T20331 CSO61T 10589936 IC50 = 66 nM T20331 CN8L4I 10590336 IC50 = 540 nM T20331 C9Q4AT 10593448 IC50 > 10000 nM T20331 CZA8K0 10596106 IC50 < 0.1 nM T20331 CAL12V 10596340 IC50 = 45 nM T20331 C3FJU2 10613667 IC50 = 30 nM T20331 CL05XO 10614625 IC50 = 1300 nM T20331 CF0H4C 10616756 IC50 = 11 nM T20331 CF3K5O 10617383 IC50 = 29 nM T20331 CU7Z2L 10617610 IC50 = 1600 nM T20331 CN0AE7 10618696 IC50 < 0.1 nM T20331 C0FP2G 10619067 Ki > 10000 nM T20331 CZ0U1P 10625004 Ki > 10000 nM T20331 CW7U9J 10637486 IC50 = 7200 nM T20331 C4J0NX 10638643 IC50 = 220 nM T20331 C24NUO 10639971 IC50 = 560 nM T20331 CI97DB 10640471 IC50 = 5100 nM T20331 CN7U4J 10641357 IC50 = 730 nM T20331 COU9W0 10642052 IC50 = 74 nM T20331 C2J8SH 10642181 IC50 = 41 nM T20331 CPI1C7 10644957 IC50 = 420 nM T20331 CFC8X2 10645176 IC50 = 670 nM T20331 C4YVF7 10645275 IC50 = 170 nM T20331 CUM24G 10662967 IC50 = 2.2 nM T20331 C7YZ5S 10664487 IC50 = 100 nM T20331 CR9U5H 10666064 IC50 = 280 nM T20331 C8CD3Y 10667042 IC50 = 730 nM T20331 CB94CS 10667094 IC50 = 4000 nM T20331 C81XIE 10668485 IC50 < 0.1 nM T20331 C3L6TA 10671331 Ki > 10000 nM T20331 C7MC2O 10672357 Ki > 10000 nM T20331 CT7XC5 10685135 IC50 = 1.2 nM T20331 C84ZVD 10685661 IC50 = 57 nM T20331 CCE0J7 10688707 IC50 = 53 nM T20331 C2P8VM 10689108 IC50 = 8.5 nM T20331 C6HQ1X 10692519 Ki > 10000 nM T20331 CDB49U 10712643 IC50 = 0.3 nM T20331 C2H8EW 10714258 IC50 = 580 nM T20331 C1MYC0 10715854 IC50 = 4000 nM T20331 C3ZVT9 10734658 IC50 = 8500 nM T20331 C9W8DT 10736124 IC50 = 0.5 nM T20331 C20VLY 10736625 IC50 = 1500 nM T20331 CPJQ74 10737530 IC50 = 79 nM T20331 CVCY89 10737532 IC50 < 0.1 nM T20331 CEQ17G 10738836 IC50 = 140 nM T20331 C0MGW2 10757242 IC50 = 10 nM T20331 CIX28F 10758195 IC50 = 910 nM T20331 C3AWR8 10758227 IC50 = 0.2 nM T20331 CON7B3 10779945 IC50 = 8200 nM T20331 C96UND 10779946 IC50 = 1200 nM T20331 C6T8XZ 10783032 IC50 > 10000 nM T20331 CU34JG 10783815 IC50 = 0.3 nM T20331 C5I4OM 10786956 IC50 = 0.7 nM T20331 C28LZT 10789271 IC50 = 8500 nM T20331 C3OD2S 10805667 IC50 = 190 nM T20331 CSY7W9 10807285 IC50 = 3 nM T20331 C71DZX 10808680 IC50 = 660 nM T20331 CR54UP 10810223 IC50 = 150 nM T20331 C8U6XP 10810784 IC50 = 2500 nM T20331 CS4JF0 10820168 Ki = 5080 nM T20331 CEH6O1 10820196 Ki = 7100 nM T20331 COER76 10830247 IC50 = 150 nM T20331 C1CPX8 10831203 IC50 = 20 nM T20331 C2B9GE 10831332 IC50 = 250 nM T20331 C2SK1O 10832634 IC50 = 380 nM T20331 C79IXY 10833009 IC50 = 460 nM T20331 CJH85Z 10833804 IC50 = 590 nM T20331 CR4S8H 10848957 IC50 = 3100 nM T20331 C7SF2X 10849420 IC50 = 160 nM T20331 CP18TD 10860014 IC50 = 230 nM T20331 CCS4J7 10872140 IC50 = 317 nM T20331 CGT23W 10872843 IC50 = 20 nM T20331 CXKT35 10883239 IC50 = 15 nM T20331 CTYL38 10892838 IC50 = 33 nM T20331 CE68CY 10892960 Ki = 62 nM T20331 CYL04M 10893873 IC50 = 78 nM T20331 C3AV8S 10903122 IC50 = 2900 nM T20331 C9IEJ1 10915401 IC50 = 0.5 nM T20331 CFHD79 10915843 IC50 < 0.1 nM T20331 C3QX4J 10916153 IC50 = 1230 nM T20331 CDMB60 10916418 IC50 < 0.1 nM T20331 CVSY25 10926406 IC50 = 1 nM T20331 CZS0V4 10926986 IC50 = 770 nM T20331 C21PAY 10927348 IC50 = 0.9 nM T20331 C6Q5FZ 10935409 IC50 = 24 nM T20331 COEM27 10947900 IC50 > 10000 nM T20331 CF8CR1 10948789 IC50 = 7500 nM T20331 CJ0OF1 10949261 IC50 < 0.1 nM T20331 C6HIZ7 10958843 IC50 = 700 nM T20331 C4QUT3 10959285 IC50 = 163 nM T20331 CM54HE 10959710 IC50 = 4 nM T20331 CFHX56 10959714 IC50 = 1307 nM T20331 C5ENC2 10969426 IC50 > 1000 nM T20331 CJT7C6 10969955 IC50 = 2 nM T20331 CT20YX 10970192 IC50 = 2 nM T20331 CPNG50 10970274 Ki = 10 nM T20331 COLK67 10970360 IC50 = 2200 nM T20331 C0YC2A 10970790 IC50 = 9500 nM T20331 CY08VU 10971233 IC50 = 70 nM T20331 C08VWM 10971892 IC50 = 8 nM T20331 CPU8M9 10981271 IC50 = 5000 nM T20331 CO98AV 10982716 IC50 = 4 nM T20331 CI6W3N 10993145 IC50 < 0.1 nM T20331 CZ31KI 11001068 IC50 = 4500 nM T20331 CFGQ04 11002751 IC50 = 3 nM T20331 C0D3VR 11002935 IC50 = 47 nM T20331 C8LMZ1 11002986 Ki = 33 nM T20331 C7Q8AJ 11003662 IC50 > 10000 nM T20331 CC28EA 11003942 IC50 = 350 nM T20331 CGSF91 11013840 IC50 = 3.1 nM T20331 C6ZSN8 11014171 IC50 = 34 nM T20331 CG20KQ 11014203 IC50 > 1000 nM T20331 C10NLV 11015360 IC50 = 8 nM T20331 C1ICL8 11025578 IC50 < 0.1 nM T20331 CHJ07Z 11035908 IC50 = 390 nM T20331 C9TVD5 11056043 IC50 = 803 nM T20331 CDK74L 11057532 Ki = 92 nM T20331 C4UPT2 11057893 IC50 = 9 nM T20331 CH2I4X 11067876 IC50 = 3400 nM T20331 CZM9I3 11068453 IC50 = 1650 nM T20331 C1JS9Y 11068838 IC50 = 507 nM T20331 CJ5EQ3 11078256 Ki = 120 nM T20331 CML5G0 11078514 IC50 = 35 nM T20331 CZR98N 11078551 IC50 > 1000 nM T20331 CGMB36 11079077 IC50 = 71 nM T20331 CEF1V3 11089837 IC50 = 710 nM T20331 C2CSO5 11099807 Ki = 450 nM T20331 C9G2RC 11099994 IC50 = 800 nM T20331 C5K2GA 11100116 IC50 > 1000 nM T20331 C2H9UY 11110676 IC50 = 2250 nM T20331 CB2E7T 11110677 IC50 = 440 nM T20331 CNMS54 11111618 IC50 = 9500 nM T20331 CW4P1L 11111992 IC50 = 1 nM T20331 C7NZV5 11130476 Ki = 260 nM T20331 CKC6D3 11133371 IC50 = 5 nM T20331 CGB78V 11143423 IC50 = 270 nM T20331 C24JXQ 11204090 IC50 = 31 nM T20331 CEF57S 11224238 IC50 = 1.8 nM T20331 CCWK17 11284878 IC50 = 120 nM T20331 CR1K5W 11342160 IC50 = 8900 nM T20331 CGM1O5 11349780 IC50 = 0.89 nM T20331 CHN8R7 11407098 IC50 = 0.92 nM T20331 C61TRZ 11491176 IC50 = 1.259 nM T20331 C2H0LY 11509561 IC50 = 3.9 nM T20331 CA69MC 11633103 IC50 = 1.8 nM T20331 CQ49SB 11640844 Ki = 5978 nM T20331 CG72WE 11727519 IC50 = 443 nM T20331 CAN06Q 11728519 IC50 > 10000 nM T20331 C7OUV9 11729353 Ki = 2.8 nM T20331 C1YWG5 11732188 IC50 < 0.1 nM T20331 C0Z9WK 11742181 Ki = 3.6 nM T20331 C8LI9U 11757324 IC50 = 23 nM T20331 C15OPT 11758930 Ki = 80 nM T20331 C43LHB 11760541 IC50 < 0.1 nM T20331 C0BM9D 11760542 IC50 < 0.1 nM T20331 C8HX1J 11781068 IC50 > 10000 nM T20331 CV5HE9 11783658 IC50 = 12 nM T20331 CR80HC 11792487 IC50 = 2600 nM T20331 CTAQ91 11792636 IC50 = 5.3 nM T20331 CMSK51 11793187 IC50 = 0.4 nM T20331 C18ERL 11795098 IC50 = 750 nM T20331 CJ5TE0 11798404 Ki > 10000 nM T20331 CY8QK9 11811424 IC50 = 282 nM T20331 CLCU02 11824465 IC50 = 3 nM T20331 CU94PX 11824961 IC50 = 127 nM T20331 C30RPC 11825270 IC50 = 380 nM T20331 CHA6Q4 12018678 IC50 > 3000 nM T20331 C3O8PX 12018679 IC50 = 79 nM T20331 C8MG7K 12018680 IC50 = 74 nM T20331 CUM43R 12071667 IC50 = 1.8 nM T20331 CY17IU 12078328 IC50 = 2400 nM T20331 CD1NO6 12078329 IC50 = 860 nM T20331 C3RJI0 12108781 IC50 = 0.97 nM T20331 CS04DT 12108783 IC50 = 1.3 nM T20331 C7FCN3 12250898 Ki = 1449 nM T20331 CV2YW1 12250899 Ki = 525 nM T20331 CM72KO 12250900 Ki = 1527 nM T20331 CO82HM 12822578 IC50 = 160 nM T20331 CVC74R 13152287 IC50 = 1800 nM T20331 C07CWK 15940921 IC50 = 2.3 nM T20331 CSI68G 17965215 IC50 = 17 nM T20331 CO7H8G 18004890 IC50 = 3.4 nM T20331 C2K0EF 18004891 IC50 = 2 nM T20331 C20CKM 18004895 IC50 = 0.57 nM T20331 C2V4FJ 18004896 IC50 = 0.85 nM T20331 CX5C4W 18004920 IC50 = 3 nM T20331 C7L4RK 18004934 IC50 = 2.7 nM T20331 CG83RC 18004938 IC50 = 3 nM T20331 CV5X0I 18004939 IC50 = 0.86 nM T20331 CQ3V2X 18004942 IC50 = 5 nM T20331 C9AL3C 18004944 IC50 = 1.3 nM T20331 CQYJ43 18004955 IC50 = 0.96 nM T20331 C6AJ8G 18004956 IC50 = 0.2 nM T20331 C9T3YH 18004985 IC50 = 1.5 nM T20331 CB28DY 18004995 IC50 = 4 nM T20331 CU06SE 18004996 IC50 = 3.3 nM T20331 C9RU0O 18004997 IC50 = 0.82 nM T20331 CPB6K0 18005004 IC50 = 2 nM T20331 C3MQC2 18735143 IC50 = 45 nM T20331 C3D2LV 20556258 IC50 = 1400 nM T20331 CA5YV8 20587799 IC50 = 9.2 nM T20331 CIYU59 20587808 IC50 = 1.5 nM T20331 CN5T3J 20610103 Ki = 52 nM T20331 C1BWC0 20610104 Ki = 303 nM T20331 C2MJI9 20610110 Ki = 88 nM T20331 CZMY80 20610111 Ki = 312 nM T20331 C5CHX2 20610116 Ki = 164 nM T20331 CMC6Q1 20610117 Ki = 819 nM T20331 CYZ21O 20610118 Ki = 130 nM T20331 C2V3AR 20610119 Ki = 799 nM T20331 CF8EY9 20647087 Ki = 109 nM T20331 C9H6AT 20647089 Ki = 1.8 nM T20331 C3KIA8 20647090 Ki = 803 nM T20331 C4ERT6 20647096 Ki = 8 nM T20331 C8K4EG 20647101 Ki = 1.9 nM T20331 CC8WN0 20647107 Ki = 19 nM T20331 CGOM78 20647122 Ki = 150 nM T20331 CM5I3B 20647123 Ki = 31 nM T20331 C5RBA6 20651572 IC50 = 3.9 nM T20331 C6TJ3X 20651581 IC50 = 1.9 nM T20331 CM37XZ 20651605 Ki = 46 nM T20331 CASE53 20651606 Ki = 2.4 nM T20331 C4ONP0 20651616 Ki = 6.7 nM T20331 COR4F2 21031286 Ki = 3.6 nM T20331 C4Q8KN 21129772 IC50 = 80000 nM T20331 CI86LK 21336486 Ki = 231 nM T20331 CO4C3S 21336489 Ki = 10 nM T20331 CT4PH1 21336493 Ki = 14 nM T20331 CW92BC 21336495 Ki = 28 nM T20331 CT7I6J 21336500 Ki = 17 nM T20331 C8VR6Y 21336503 Ki = 26 nM T20331 CH19JC 21336507 Ki = 10 nM T20331 C89KZL 21336511 Ki = 11 nM T20331 CIL9Q8 21956072 IC50 = 7.7 nM T20331 CD48GB 22253974 IC50 = 0.6 nM T20331 CL4F7O 22254003 IC50 = 10.4 nM T20331 CEOA23 22254020 Ki = 1.9 nM T20331 CBS20U 22254050 Ki = 2.8 nM T20331 CO32YX 22254068 Ki = 1.5 nM T20331 C74ZCP 22254110 Ki = 1.7 nM T20331 C82IGT 22254119 Ki = 13.9 nM T20331 CHQT84 22254131 Ki = 4.9 nM T20331 C6CQS8 22257112 IC50 = 91 nM T20331 CCL3I8 22257113 IC50 = 111 nM T20331 CA70RF 22288540 Ki = 385 nM T20331 C5V7MW 22325320 IC50 = 4.8 nM T20331 CVUF07 22325323 IC50 = 28 nM T20331 CO9QJ1 22325333 IC50 = 5.7 nM T20331 CP7E2N 22325336 IC50 = 6.6 nM T20331 CN4Z6U 22325338 IC50 = 37 nM T20331 CXC31N 22325344 IC50 = 140 nM T20331 CZ8AS7 22325346 IC50 = 36 nM T20331 CU3RJ9 22325347 IC50 = 51 nM T20331 CRJC06 22325349 IC50 > 1000 nM T20331 C9L7IT 22325350 IC50 = 85 nM T20331 C6HD2P 22458796 Ki = 11 nM T20331 CH7D8V 22458799 Ki = 4.7 nM T20331 C4GJH6 22458813 Ki = 0.84 nM T20331 CT58QA 22458823 Ki = 3.4 nM T20331 C0PB4U 22462213 Ki = 46 nM T20331 CV43SE 22639804 IC50 = 6 nM T20331 CE46QI 22660756 IC50 = 2.1 nM T20331 C1G7TQ 22934114 IC50 = 13 nM T20331 CLA5C6 22934115 IC50 = 110 nM T20331 C5LF6H 22934118 IC50 = 6.4 nM T20331 CD19NL 22934120 IC50 = 110 nM T20331 CV76TJ 22934124 IC50 = 5.8 nM T20331 CJW92R 22934127 IC50 = 7.3 nM T20331 CIEJ92 22934129 IC50 = 20 nM T20331 C91KPN 22934130 IC50 = 25 nM T20331 C1Q6HI 22934131 IC50 = 46 nM T20331 CB3VZ1 22934132 IC50 = 2.3 nM T20331 CQ4YA2 22934136 IC50 = 6.3 nM T20331 C54UYQ 22934142 IC50 = 6.4 nM T20331 CN6HU8 22934144 IC50 = 32 nM T20331 CI2UW8 23283651 IC50 = 337 nM T20331 C7H4GQ 23283663 IC50 = 7 nM T20331 C0WKZ6 23283666 IC50 = 443 nM T20331 CQ4SF7 23397122 Ki = 2165 nM T20331 C43HJL 24987242 Ki = 1.995 nM T20331 CN5S1B 24994659 Ki = 0.03162 nM T20331 CYJW69 24996879 Ki = 0.07943 nM T20331 CKR94M 25022356 Ki = 316.23 nM T20331 CG3VL7 25067562 IC50 = 3.3 nM T20331 COE3T5 25071310 Ki = 0.3162 nM T20331 CUK64D 25071620 Ki = 0.1995 nM T20331 CZ48AL 25071621 Ki = 0.1585 nM T20331 C6I7JN 25071929 Ki = 1.259 nM T20331 CFE62W 25071930 Ki = 19.95 nM T20331 CU0SR4 25071931 Ki = 0.631 nM T20331 C18XGM 25072242 Ki = 1.585 nM T20331 CR75FH 25072243 Ki = 5.012 nM T20331 CG71VR 25072244 Ki = 19.95 nM T20331 C8QW3Y 25072245 Ki = 2.512 nM T20331 C4RE0M 25072246 Ki = 25.12 nM T20331 CTWZ82 25072568 Ki = 79.43 nM T20331 CW2H9F 25072875 Ki = 0.3981 nM T20331 CA4FV9 25072876 Ki = 5.012 nM T20331 CPUB18 25072877 Ki = 0.631 nM T20331 C6GPL3 25072880 Ki = 0.3162 nM T20331 CDY9Z4 25073188 Ki = 7.943 nM T20331 C3AJD0 25073189 Ki = 0.631 nM T20331 C9KR8V 25073190 Ki = 0.3162 nM T20331 C68FHZ 25073191 Ki = 1.259 nM T20331 C98ISN 25073801 Ki = 1.259 nM T20331 CB9O5E 25074110 Ki = 3.981 nM T20331 C7IH3J 25181112 Ki > 2000 nM T20331 C7VID1 25211875 IC50 = 7.2 nM T20331 CNU7P4 42630820 Ki = 1.3 nM T20331 C7GSL3 44138575 Ki = 145 nM T20331 CSM1A0 44138577 Ki = 2.6 nM T20331 C4VYG8 44138579 Ki = 1.9 nM T20331 C3WOD7 44138581 Ki = 2.5 nM T20331 C4P8OL 44138706 Ki = 1 nM T20331 CW2G7S 44138708 Ki = 1.8 nM T20331 C7H3NP 44138709 Ki = 1.4 nM T20331 CU4XB0 44139234 Ki = 1 nM T20331 CFX6J1 44139354 Ki = 300 nM T20331 CDF14X 44139355 Ki = 8.6 nM T20331 C4Q9IL 44139356 Ki = 3.1 nM T20331 CG3KU0 44139478 Ki = 1.6 nM T20331 CXR3J2 44139479 Ki = 0.8 nM T20331 CW8J0K 44139480 Ki = 3.2 nM T20331 COJK15 44139481 Ki = 5.9 nM T20331 CX17RC 44139599 Ki = 2.5 nM T20331 CY0GQ3 44139600 Ki = 5.1 nM T20331 CVCH41 44139601 Ki = 2.2 nM T20331 C79OCX 44139602 Ki = 2 nM T20331 C9Z0RV 44139603 Ki = 4.1 nM T20331 C2U9ES 44139732 Ki = 1.1 nM T20331 CNER41 44158441 Ki = 5.012 nM T20331 CM9X7F 44158542 Ki = 0.02512 nM T20331 C6JU4Z 44158545 Ki = 0.3162 nM T20331 CW3L6N 44158762 Ki = 0.0631 nM T20331 CHQI47 44158763 Ki = 0.1 nM T20331 CS2P6L 44158764 Ki = 0.0631 nM T20331 C8XTC1 44159235 Ki = 1 nM T20331 C17DRZ 44159236 Ki = 0.1585 nM T20331 CCF83L 44159353 Ki = 0.1585 nM T20331 CL2T0G 44159473 Ki = 0.1259 nM T20331 C36WFY 44159706 Ki = 1.585 nM T20331 CXG52N 44160199 Ki = 0.3162 nM T20331 C3KE4D 44160200 Ki = 0.2512 nM T20331 CLX51J 44249749 Ki > 10000 nM T20331 CA97BE 44263876 IC50 = 52 nM T20331 C5TSD8 44263987 IC50 = 570 nM T20331 CWY4I3 44264067 IC50 = 6100 nM T20331 C1ZU9V 44271202 IC50 = 0.7 nM T20331 CQME72 44271207 IC50 = 0.85 nM T20331 CY74TA 44271208 IC50 = 3.3 nM T20331 CV7JF5 44271223 IC50 = 1.1 nM T20331 C5A0CN 44271231 IC50 = 6.1 nM T20331 CXQ18V 44271267 IC50 = 1.7 nM T20331 C5U2AE 44271276 IC50 = 0.59 nM T20331 CK63LT 44271284 IC50 = 1.4 nM T20331 CY32KS 44271289 IC50 = 1.3 nM T20331 CPQ82N 44271317 IC50 = 1.4 nM T20331 C30PUR 44271318 IC50 = 4.7 nM T20331 C80NPO 44271355 IC50 = 2.8 nM T20331 C0YT5C 44271373 IC50 = 2.3 nM T20331 C94IFM 44271377 IC50 = 4.4 nM T20331 CQ2DE3 44271382 IC50 = 0.71 nM T20331 CA83FE 44271385 IC50 = 0.89 nM T20331 CI2OV0 44271437 IC50 = 710 nM T20331 CG89EY 44271442 IC50 = 110 nM T20331 C2O0JK 44271450 IC50 = 200 nM T20331 C2IR6Y 44271459 IC50 = 100 nM T20331 CT4J7P 44271460 IC50 = 210 nM T20331 CX93WE 44271463 IC50 = 2000 nM T20331 C63FGN 44271467 IC50 = 510 nM T20331 CY3U9A 44271468 IC50 = 310 nM T20331 CN6SY4 44271478 IC50 = 4 nM T20331 CM4DU9 44271482 IC50 = 51 nM T20331 CCKY51 44271484 IC50 = 290 nM T20331 CL1PF9 44271486 IC50 = 38 nM T20331 CCB80J 44271487 IC50 = 4 nM T20331 CM2E8D 44271493 IC50 = 16 nM T20331 CIM1F9 44271506 IC50 = 33 nM T20331 C6ITF7 44271517 IC50 = 20 nM T20331 C0FDP8 44271525 IC50 = 390 nM T20331 CL28IN 44271529 IC50 = 380 nM T20331 CX1AN3 44271531 IC50 = 2.9 nM T20331 CSI1W8 44271532 IC50 = 270 nM T20331 C7Y0XG 44271533 IC50 = 58 nM T20331 CAR4Y6 44271541 IC50 = 250 nM T20331 CNW12L 44271542 IC50 = 0.9 nM T20331 C2T6CH 44271549 IC50 = 2 nM T20331 CP48BY 44271550 IC50 = 33 nM T20331 CJL24X 44271556 IC50 = 1000 nM T20331 CP4K6A 44271559 IC50 = 0.6 nM T20331 CEI0R2 44271562 IC50 = 4900 nM T20331 C92TCK 44271565 IC50 = 2.7 nM T20331 CRV9I7 44271592 IC50 = 46 nM T20331 C0SF7N 44271637 IC50 = 44 nM T20331 C9FV7D 44271638 IC50 = 400 nM T20331 C28IWX 44271691 IC50 = 50 nM T20331 C6KR1Y 44287938 IC50 = 770 nM T20331 CHT17W 44287971 IC50 = 68000 nM T20331 C2IXS5 44287982 IC50 = 163000 nM T20331 C7X5DG 44287999 IC50 = 48000 nM T20331 C1FW4N 44288067 IC50 = 25000 nM T20331 CAI9T7 44288112 IC50 = 75000 nM T20331 CN76WT 44288390 IC50 = 2600 nM T20331 CS1FG8 44288395 IC50 = 11900 nM T20331 CHI04U 44289698 IC50 = 16 nM T20331 C30YQX 44289816 IC50 = 114 nM T20331 C8XLO5 44289818 IC50 = 31 nM T20331 C8UQ1V 44289827 IC50 = 39 nM T20331 C8H1UF 44289833 IC50 = 140 nM T20331 CY6O2J 44289834 IC50 = 17 nM T20331 CR17GO 44289857 IC50 = 170 nM T20331 C4Q3OV 44289890 IC50 = 26 nM T20331 C34VAI 44289909 IC50 = 30 nM T20331 CFI24H 44294739 Ki = 724 nM T20331 CY4O0T 44294740 Ki = 151 nM T20331 C5Y7HO 44294762 Ki = 103 nM T20331 CMP3F8 44294789 Ki = 724 nM T20331 CTM0K1 44294898 Ki = 4120 nM T20331 CZV6U3 44294942 Ki = 123 nM T20331 C0Y5UT 44294983 Ki = 412 nM T20331 CJ8BK4 44295007 Ki = 199 nM T20331 CI6O2E 44295107 Ki = 426 nM T20331 CV74NB 44295115 Ki = 95 nM T20331 CCT79B 44295138 Ki = 724 nM T20331 C9YMC7 44295140 Ki > 100000 nM T20331 CNV3D1 44302732 Ki = 0.3 nM T20331 C01TMJ 44308120 IC50 > 1000 nM T20331 CF83NV 44308516 IC50 = 121 nM T20331 CL3V4F 44312687 IC50 = 709 nM T20331 COP85Y 44312689 IC50 > 1000 nM T20331 C53NZM 44312707 IC50 = 487 nM T20331 C9HU8I 44312735 IC50 > 1000 nM T20331 C8W2XK 44312754 IC50 = 20 nM T20331 C1WGX9 44312757 IC50 > 1000 nM T20331 CY93CN 44312759 IC50 > 1000 nM T20331 CR4LW1 44312780 IC50 = 10 nM T20331 CKX72U 44312926 IC50 = 37 nM T20331 CM8P3X 44312927 IC50 = 436 nM T20331 CLEZ60 44312955 IC50 = 29 nM T20331 CI7J0S 44312956 IC50 = 67 nM T20331 C67USH 44312965 IC50 = 114 nM T20331 C2KEC1 44312968 IC50 = 63 nM T20331 C8UWM3 44312976 IC50 > 3000 nM T20331 C6XNJ4 44312981 IC50 = 40 nM T20331 C0JGE6 44313039 IC50 = 303 nM T20331 C1AHN7 44313042 IC50 = 37 nM T20331 CQD95S 44313057 IC50 = 229 nM T20331 CGKD32 44313061 IC50 = 178 nM T20331 COGA86 44313076 IC50 > 1000 nM T20331 C4JLP3 44313078 IC50 = 145 nM T20331 C7I2JZ 44313092 IC50 = 162 nM T20331 C2TR0N 44313099 IC50 = 48 nM T20331 CXI23J 44313223 IC50 = 359 nM T20331 C51LQV 44313224 IC50 = 520 nM T20331 CQO28I 44313228 IC50 = 763 nM T20331 CMJ6X1 44313241 IC50 = 267 nM T20331 C20RSX 44313274 IC50 = 356 nM T20331 C8KY4W 44313308 IC50 > 1000 nM T20331 CUZ46W 44313310 IC50 > 1000 nM T20331 CZY39A 44313318 IC50 > 1000 nM T20331 C06CFY 44313331 IC50 = 100 nM T20331 CJ2A8C 44313362 IC50 > 1000 nM T20331 C7Y6QL 44313363 IC50 > 1000 nM T20331 C3JRL1 44313486 IC50 = 670 nM T20331 CD1MK7 44313494 IC50 = 292 nM T20331 CGJO91 44313495 IC50 = 573 nM T20331 CYU8M3 44313496 IC50 = 759 nM T20331 CSG9Q0 44313505 IC50 > 1000 nM T20331 CF79IP 44313510 IC50 = 622 nM T20331 CLNX65 44313529 IC50 > 1000 nM T20331 CW3HQ1 44313570 IC50 = 233 nM T20331 C3SA4G 44313571 IC50 > 1000 nM T20331 C3L4WV 44313572 IC50 = 800 nM T20331 C4H8UO 44313576 IC50 = 197 nM T20331 CR19HQ 44313594 IC50 > 1000 nM T20331 C10LCM 44313595 IC50 > 1000 nM T20331 CM3C8J 44313596 IC50 = 431 nM T20331 CK5FP6 44344208 IC50 = 27 nM T20331 C2JY7D 44344243 IC50 = 1 nM T20331 C2YO4X 44344244 IC50 = 75 nM T20331 CN83KW 44344259 IC50 = 22 nM T20331 CBG4V3 44344283 IC50 = 53 nM T20331 CHJ6R9 44344312 IC50 = 11 nM T20331 CTG82D 44344352 IC50 = 40 nM T20331 CZVQ53 44344356 IC50 = 11 nM T20331 CQS03U 44344454 IC50 = 19 nM T20331 CDJL59 44344455 IC50 = 27 nM T20331 C3L8SQ 44344468 IC50 = 5 nM T20331 CM2F4T 44344497 IC50 = 10 nM T20331 C4D2XF 44344599 IC50 = 5 nM T20331 C7T9PV 44344608 IC50 = 12 nM T20331 CE1Q5D 44344629 IC50 = 40 nM T20331 CEX95R 44344633 IC50 = 300 nM T20331 CA65WB 44344734 IC50 = 350 nM T20331 C7IZ8K 44345637 Ki = 4769 nM T20331 C4XN2Y 44345638 Ki = 210 nM T20331 C4X0UP 44345650 Ki = 37 nM T20331 CDX3B7 44345719 Ki = 231 nM T20331 CZ6GA7 44345737 Ki = 40 nM T20331 CQ5B3P 44345744 Ki = 116 nM T20331 C3MOZ8 44345745 Ki > 10000 nM T20331 CW87CF 44345801 Ki = 4.9 nM T20331 C8LPF9 44345802 Ki = 56 nM T20331 CV6AW8 44345803 Ki = 14 nM T20331 CAT3N2 44345818 Ki = 19 nM T20331 C25AGB 44345820 Ki = 8 nM T20331 CJ46CZ 44345853 Ki = 4 nM T20331 CK0V1T 44345854 Ki = 69 nM T20331 CHE8G0 44345855 Ki = 3001 nM T20331 CA15EX 44345933 Ki = 3.5 nM T20331 C3RX1B 44345934 Ki = 30 nM T20331 CH2A8E 44345935 Ki = 34 nM T20331 C47LTV 44345940 Ki = 148 nM T20331 C5K7LN 44345949 Ki = 21 nM T20331 C4BIF1 44345961 Ki = 40 nM T20331 C2P5VT 44345971 Ki = 27 nM T20331 C4VD6X 44370176 IC50 = 42.9 nM T20331 CU73FW 44370177 IC50 = 279 nM T20331 CVN1P2 44370179 IC50 = 32.2 nM T20331 C1UQR5 44370180 IC50 = 175 nM T20331 C2D7YV 44370202 IC50 = 92.2 nM T20331 CH8QJ6 44370214 IC50 = 47.7 nM T20331 C7HF2B 44370215 IC50 = 48.4 nM T20331 CV82UW 44370240 IC50 = 20.4 nM T20331 CKGN86 44370250 IC50 = 147 nM T20331 CF65OZ 44370266 IC50 = 28.4 nM T20331 C4M5YB 44370270 IC50 = 142 nM T20331 CA1F2O 44377440 IC50 = 68 nM T20331 C8D6VU 44377450 IC50 = 45 nM T20331 CK3B4D 44377452 IC50 = 39 nM T20331 CUEY97 44377460 IC50 = 79 nM T20331 C87OLK 44377461 IC50 = 72 nM T20331 C94TQS 44377468 IC50 = 85 nM T20331 CT7KH4 44377476 IC50 = 190 nM T20331 C1S8JB 44377661 IC50 = 680 nM T20331 C6OZ2W 44377681 IC50 > 1000 nM T20331 CW32ZL 44377689 IC50 = 740 nM T20331 CQ2NH8 44377690 IC50 = 1000 nM T20331 CYW82X 44377691 IC50 = 52 nM T20331 CO7RQ6 44377722 IC50 = 540 nM T20331 CR0I6K 44377731 IC50 = 66 nM T20331 CPL24E 44377734 IC50 = 210 nM T20331 C0TK1X 44377854 IC50 = 86 nM T20331 CD43BA 44377915 IC50 = 310 nM T20331 C4TGV7 44377916 IC50 = 140 nM T20331 C2C6YP 44379085 IC50 = 3.7 nM T20331 C5PLS6 44379089 IC50 = 13 nM T20331 C39RNP 44379095 IC50 = 1.2 nM T20331 CU97WP 44379101 IC50 = 1 nM T20331 C5B0UL 44379102 IC50 = 28 nM T20331 CVTE78 44379363 IC50 = 24 nM T20331 CTH68M 44379364 IC50 = 56 nM T20331 CZ2Y3E 44379410 IC50 = 11 nM T20331 CUS3I7 44379411 IC50 = 66 nM T20331 CE25YT 44390369 IC50 = 460 nM T20331 CFH3C2 44390385 IC50 = 560 nM T20331 C6LJC2 44390456 IC50 > 1000 nM T20331 CHGY52 44390499 IC50 = 470 nM T20331 CPQ63J 44390733 IC50 > 1000 nM T20331 C3TEB2 44390752 IC50 > 1000 nM T20331 C4RN8A 44401449 IC50 = 880 nM T20331 C49USD 44401460 IC50 = 41 nM T20331 CHGX51 44401508 IC50 = 4.9 nM T20331 CIKD90 44401552 IC50 = 78 nM T20331 C8VQ3B 44401591 IC50 = 1.6 nM T20331 CT46VH 44401616 IC50 = 2.5 nM T20331 CIXE76 44401626 IC50 = 120 nM T20331 CER15G 44401671 IC50 = 3000 nM T20331 CPV72O 44453965 Ki = 405 nM T20331 CV06JE 44460453 IC50 = 5 nM T20331 C3JZM2 44460467 IC50 = 7 nM T20331 CSH61O 44460473 IC50 = 17 nM T20331 CJR6A9 44460506 IC50 = 71 nM T20331 C8S2UW 44460681 IC50 = 20 nM T20331 CM0LX7 44460704 IC50 = 21 nM T20331 C5MVL6 44460707 IC50 = 19 nM T20331 CN1QB8 44460712 IC50 = 22 nM T20331 C0LF4H 44460713 IC50 = 37 nM T20331 CGZ10A 44460788 IC50 = 18 nM T20331 C25BTF 44460789 IC50 = 41 nM T20331 CN68MR 44460798 IC50 = 25 nM T20331 CB21OZ 44460811 IC50 = 15 nM T20331 C6Z7QR 44460812 IC50 = 2460 nM T20331 CBXJ80 44460815 IC50 = 78 nM T20331 CJQ2K5 44460830 IC50 = 25 nM T20331 CWH36L 44460842 IC50 = 23 nM T20331 C4N9KT 44460868 IC50 = 210 nM T20331 C05RLI 44460881 IC50 = 150 nM T20331 CI01LN 44460883 IC50 = 29 nM T20331 CEM6X7 44460907 IC50 = 6 nM T20331 C0QU9W 44460919 IC50 = 2 nM T20331 C0U5LD 44460920 IC50 = 4 nM T20331 CSF8V7 44460921 IC50 = 81 nM T20331 CH9YC0 44460922 IC50 = 18 nM T20331 CVA6T2 44460943 IC50 = 15 nM T20331 CTD54R 44460946 IC50 = 7 nM T20331 C20BYE 44460957 IC50 = 6 nM T20331 CQR19W 44460963 IC50 = 6 nM T20331 CN9X1R 44460964 IC50 = 290 nM T20331 C7CN2P 44460972 IC50 = 5 nM T20331 CNF7M5 44460988 IC50 = 2 nM T20331 C67ERA 44461003 IC50 = 15 nM T20331 C7G6YQ 44461006 IC50 = 4 nM T20331 C51HNI 44461018 IC50 = 3 nM T20331 CXSD35 44461022 IC50 = 2 nM T20331 CHW5C6 44461023 IC50 = 1 nM T20331 CD8XE9 44461040 IC50 = 40 nM T20331 CFMD78 44461051 IC50 = 2 nM T20331 CDT52L 44461106 IC50 = 99 nM T20331 C8SV0A 44461107 IC50 = 13 nM T20331 CJM96N 44461116 IC50 = 5 nM T20331 CFOL91 44461118 IC50 = 20 nM T20331 CCD0R2 44461145 IC50 = 38 nM T20331 CD0OS8 44461159 IC50 = 17 nM T20331 C9J7TX 44461179 IC50 = 6 nM T20331 CP98UG 44461180 IC50 = 2 nM T20331 C9FJ5R 44461196 IC50 = 3 nM T20331 CXIB36 44461198 IC50 = 6 nM T20331 CY05KT 44461199 IC50 = 3 nM T20331 C9IPG8 44461200 IC50 = 2 nM T20331 CG1XA8 44461201 IC50 = 15 nM T20331 C3VOY4 44461208 IC50 = 6 nM T20331 CXN52U 44461210 IC50 = 6 nM T20331 CX10TB 44573407 IC50 = 32 nM T20331 CB67TW 44573408 IC50 = 630 nM T20331 C81LSB 44573448 IC50 = 130 nM T20331 CB2N9P 44573449 IC50 = 160 nM T20331 CST40L 44573531 IC50 = 44 nM T20331 CZ9L3W 44573532 IC50 = 270 nM T20331 C2OKR6 44573533 IC50 = 59 nM T20331 CEW06D 44573534 IC50 = 51 nM T20331 CD51BH 44573541 IC50 = 1.4 nM T20331 C4F8JE 44573565 IC50 = 300 nM T20331 C5TGX9 44573566 IC50 > 1000 nM T20331 CKNF08 44573567 IC50 = 160 nM T20331 C0ET9R 44573574 IC50 = 1.2 nM T20331 CM1US2 44573575 IC50 = 7.5 nM T20331 C0PT1H 44573606 IC50 = 160 nM T20331 C30WFC 44573607 IC50 = 350 nM T20331 CGN71L 44573614 IC50 = 23 nM T20331 CD0AK9 44573615 IC50 = 9.8 nM T20331 C07EAQ 44573616 IC50 = 430 nM T20331 CNP27R 44573646 IC50 = 39 nM T20331 CZ40VS 44573647 IC50 = 17 nM T20331 C9NV2T 44573648 IC50 = 4.8 nM T20331 CNW60R 44573656 IC50 = 180 nM T20331 CSG8A4 44573697 IC50 = 8.1 nM T20331 C2IB3G 44573704 IC50 = 3 nM T20331 C5WF4I 44573705 IC50 = 2.1 nM T20331 CSRQ65 44573743 IC50 = 3 nM T20331 CN4J3K 44579794 IC50 = 91 nM T20331 CBJ9W6 44579806 IC50 = 20 nM T20331 CON7W6 44579807 IC50 = 39 nM T20331 CYR94Z 44579808 IC50 = 47 nM T20331 CI5Y8R 44579809 IC50 = 45 nM T20331 CLM42D 44579810 IC50 = 2.3 nM T20331 C1KSB8 44579825 IC50 = 2.4 nM T20331 CH03CS 44579826 IC50 = 2.4 nM T20331 CUV47M 44579827 IC50 = 3.1 nM T20331 CY9Z5J 44579845 IC50 = 8 nM T20331 C6YR0Q 44579846 IC50 = 2.2 nM T20331 CV4D5I 44579847 IC50 > 1000 nM T20331 C0DC9S 44579862 IC50 = 2.2 nM T20331 C2E6CF 44579863 IC50 = 4.5 nM T20331 CVE3C0 44579864 IC50 = 15 nM T20331 CZ65XF 44579887 IC50 = 5.1 nM T20331 C1ONS7 44579888 IC50 = 2.1 nM T20331 CVO10S 44580050 IC50 = 1.4 nM T20331 CV37ED 44580100 IC50 = 6.7 nM T20331 COCM85 44580222 IC50 = 9.3 nM T20331 CQ5U4M 44580223 IC50 = 2.2 nM T20331 CGPE10 44580463 IC50 > 1000 nM T20331 CKP9M4 44580502 IC50 = 10000 nM T20331 C2IK8H 44580503 IC50 = 1600 nM T20331 C3FU8S 44580504 IC50 = 4900 nM T20331 C5VC7D 44580505 IC50 = 91 nM T20331 C7P9VE 44580546 IC50 = 500 nM T20331 CJ1D6U 44580547 IC50 = 74 nM T20331 C5A6WX 44580593 IC50 = 250 nM T20331 CZ5YD2 44580594 IC50 = 83 nM T20331 CQ6BH5 44580665 IC50 = 17 nM T20331 C1EVY0 44580666 IC50 = 10 nM T20331 C1XE2D 44580667 IC50 = 10 nM T20331 CF9M7V 44580708 IC50 = 1.8 nM T20331 CCM6Z3 44580709 IC50 = 2 nM T20331 C3Y4PC 44580710 IC50 = 110 nM T20331 C0K5MI 44580745 IC50 = 20 nM T20331 C26SNF 44580746 IC50 = 58 nM T20331 CX4W5U 44580747 IC50 = 130 nM T20331 CHD45B 44580748 IC50 = 56 nM T20331 C29QNK 44583225 IC50 > 1000 nM T20331 C5XZ6B 44583277 IC50 > 1000 nM T20331 C8PKL2 44583377 IC50 > 1000 nM T20331 CZD91P 44583378 IC50 > 1000 nM T20331 C4ZLA1 44583394 IC50 = 1.1 nM T20331 CY2IH8 44583395 IC50 = 3.9 nM T20331 C6I5FE 44583435 IC50 = 1.1 nM T20331 C1F6ZL 44583436 IC50 = 1.8 nM T20331 C09UZV 44583437 IC50 = 14 nM T20331 CYE48Q 44583438 IC50 = 0.99 nM T20331 CHA42V 44583462 IC50 = 2.4 nM T20331 C0YW3P 44583463 IC50 = 1.3 nM T20331 C09ZBL 44583505 IC50 = 20 nM T20331 C3XI5V 44583506 IC50 = 2.2 nM T20331 CD1JQ0 44583507 IC50 = 6.1 nM T20331 CK95ZB 44583539 IC50 = 0.83 nM T20331 C3A2RP 44583540 IC50 = 1 nM T20331 C9YF7J 44583541 IC50 = 0.69 nM T20331 CNA9Q8 44583556 IC50 = 2.9 nM T20331 C4ILR6 44583557 IC50 = 2.3 nM T20331 C0Z3JA 44583558 IC50 = 3.5 nM T20331 CLQ27Y 44583559 IC50 = 1.8 nM T20331 C54ZPF 44583560 IC50 = 7.9 nM T20331 C24GEC 44583588 IC50 = 3.4 nM T20331 C7PW2H 45481639 IC50 = 11 nM T20331 C9X5PM 45481640 IC50 = 7.1 nM T20331 CV4MJ1 45481641 IC50 = 2.6 nM T20331 CW1E8I 45481642 IC50 = 3.2 nM T20331 CB51KA 45481643 IC50 = 41 nM T20331 CVH43K 45481644 IC50 > 1000 nM T20331 CC05EP 45481795 IC50 = 4.1 nM T20331 CKE1A4 45481797 IC50 = 4.9 nM T20331 CZLA60 45481798 IC50 = 1.4 nM T20331 CSY29X 45481799 IC50 = 5.4 nM T20331 C6YPK8 45481800 IC50 = 2.5 nM T20331 CUX3O8 45481801 IC50 = 3.2 nM T20331 CVI10Q 45481802 IC50 = 8.9 nM T20331 C4VYT2 45481803 IC50 = 3.9 nM T20331 CS8BG4 45481804 IC50 = 2.2 nM T20331 CD38WP 45481805 IC50 = 3.4 nM T20331 CDI9A8 45481806 IC50 = 5 nM T20331 CMH1I4 45481807 IC50 = 2.4 nM T20331 CCQP02 45481808 IC50 = 4.2 nM T20331 C9ZPK5 45481809 IC50 = 1.8 nM T20331 C6WC7N 45481810 IC50 = 6.1 nM T20331 CUT3C2 45481811 IC50 = 2.8 nM T20331 C30LDO 45487447 IC50 > 10000 nM T20331 CL9PW1 45487448 IC50 > 10000 nM T20331 CMKY87 45487530 IC50 = 2.3 nM T20331 C17UHB 45487535 IC50 = 7.5 nM T20331 CYK1Z0 45487538 IC50 = 2 nM T20331 C84MXI 45487565 IC50 = 2.9 nM T20331 C16MRO 45487576 IC50 = 2.2 nM T20331 CC91ZS 45487589 IC50 = 2.2 nM T20331 CR7JB4 45487608 IC50 = 3 nM T20331 C6XD3O 45487628 IC50 = 2.2 nM T20331 CCF6A1 45487629 IC50 = 4.5 nM T20331 CV4C7O 45487630 IC50 = 3.1 nM T20331 CZ1T4R 45487631 IC50 = 2.7 nM T20331 C2CW9E 45487632 IC50 = 2.6 nM T20331 CKJ26Y 46209585 Ki = 12 nM T20331 CWK60Y 46209598 Ki = 9.2 nM T20331 CX3IA2 46226575 IC50 = 2.8 nM T20331 CI51FD 46226580 IC50 = 2.2 nM T20331 CEK9C5 46226606 IC50 = 5.4 nM T20331 CH1L9M 46226607 IC50 = 2 nM T20331 CC6V2I 46226612 IC50 = 2.7 nM T20331 CI0TN6 46226627 IC50 = 2.4 nM T20331 CB9S7A 46226628 IC50 = 2.1 nM T20331 C4A6RZ 46226635 IC50 = 2.9 nM T20331 CUB25C 46226636 IC50 = 2.4 nM T20331 C90RQC 46226641 IC50 = 1.2 nM T20331 CKIN21 46226642 IC50 = 26 nM T20331 CC4UY2 46226653 IC50 = 2.2 nM T20331 CZD7T5 46880224 Ki > 10000 nM T20331 C2V0OW 46912327 Ki = 12 nM T20331 C49PEN 46913408 Ki = 8 nM T20331 CNK46O 46913409 Ki = 5 nM T20331 C3ABO0 46913508 Ki = 6 nM T20331 CA2ND0 46913511 Ki = 8 nM T20331 CR3X6E 46913512 Ki = 9 nM T20331 CMBC38 46913606 Ki = 5 nM T20331 CYBL50 46913706 Ki = 2 nM T20331 C8GAI9 46927903 Ki = 7.943 nM T20331 CBEO38 46927904 Ki = 2511.89 nM T20331 C9PCE3 49862155 Ki = 2.512 nM T20331 CXFB82 49862156 Ki = 2.512 nM T20331 CLI2D5 49862157 Ki = 1 nM T20331 CZL84X 49862158 Ki = 1.585 nM T20331 CS29DQ 49862198 Ki = 5.012 nM T20331 CJP50V 49862199 Ki = 50.12 nM T20331 CZST43 49862200 Ki = 1 nM T20331 C6HM1T 49862239 Ki = 0.3981 nM T20331 CGA8E9 49862240 Ki = 0.7943 nM T20331 CS05YG 49862241 Ki = 0.631 nM T20331 COH7B3 49862288 Ki = 5.012 nM T20331 CX4BJ9 49862289 Ki = 0.7943 nM T20331 CS5E1Z 49862290 Ki = 5.012 nM T20331 C6EZ3P 49862336 Ki = 31.62 nM T20331 CE39XV 49862337 Ki = 1000 nM T20331 CK6NJ2 49862338 Ki = 3.981 nM T20331 CBW4D7 49862339 Ki = 1.585 nM T20331 C3DBR2 49862340 Ki = 3.981 nM T20331 CK93DQ 49862400 Ki = 0.631 nM T20331 CRD04W 49862401 Ki = 1.259 nM T20331 CGO62F 50925473 Ki > 3981.07 nM T20331 CI69YC 52941430 Ki = 0.0631 nM T20331 CETZ86 52942650 Ki = 0.1 nM T20331 CU0L2Y 52942663 Ki = 0.1 nM T20331 C26TPC 52942671 Ki = 0.1 nM T20331 C2KAG4 52943793 Ki = 0.631 nM T20331 C3QGT9 52944983 Ki = 0.03981 nM T20331 CCY08N 52948742 Ki = 0.1995 nM T20331 CNV30K 52948986 Ki = 0.1995 nM T20331 C3Z5LA 52950004 Ki = 0.1585 nM T20331 CH5A3Z 52953217 Ki > 5000 nM T20331 CV10HR 52953219 Ki > 400 nM T20331 C6Q3GO 54141274 Ki = 1.4 nM T20331 C8SW7T 54580488 Ki = 42 nM T20331 C4JNK2 54580489 Ki = 2.6 nM T20331 C94RKM 54581508 Ki = 8.6 nM T20331 C2SA5T 54582033 Ki > 1000 nM T20331 CH0E6D 54582496 Ki = 8.6 nM T20331 CQ1C4L 54583973 Ki = 7.3 nM T20331 C2MK8P 54584448 Ki = 28 nM T20331 CFLH85 54586366 Ki = 350 nM T20331 C1P2JA 54587390 Ki = 6.9 nM T20331 CZY7F9 54752621 Ki = 7.6 nM T20331 CQCK34 56659886 Ki = 200 nM T20331 CQMT25 56659887 Ki = 23 nM T20331 C15PTA 56659888 Ki = 8.4 nM T20331 C54GDV 56663345 Ki = 1.8 nM T20331 CQR19Y 56663346 Ki = 170 nM T20331 CC79DE 56663347 Ki = 370 nM T20331 CG15UN 56666777 Ki = 0.9 nM T20331 C0O5WM 56666778 Ki = 0.6 nM T20331 C7TQ1V 56666779 Ki = 0.8 nM T20331 CG6R5I 56670210 Ki = 210 nM T20331 CN87CB 56673731 Ki = 27 nM T20331 CRLC95 56673732 Ki = 420 nM T20331 C6L0PI 56673733 Ki = 60 nM T20331 CV3G9F 56673734 Ki = 14 nM T20331 CSK35M 56677038 Ki = 1900 nM T20331 C8S7RJ 56677039 Ki = 21 nM T20331 CA8LQ9 56677040 Ki = 97 nM T20331 C60SVM 56677041 Ki = 3.4 nM T20331 CMC76B 56677042 Ki = 88 nM T20331 CFPM34 56677043 Ki = 4.4 nM T20331 C06MVW 56683702 Ki = 19 nM T20331 CVJ0E7 56683703 Ki = 6.9 nM T20331 C0S3HY 56683704 Ki = 0.3 nM T20331 CY1VA4 56683705 Ki = 0.8 nM T20331 CM9JD1 56683706 Ki = 110 nM T20331 CU3NW8 56683832 IC50 = 5 nM T20331 CLQ9Y2 56841989 Ki = 0.5 nM T20331 C8CGX9 57345520 Ki = 0.5 nM T20331 CLA76G 57345521 Ki = 0.3 nM T20331 CFMT71 57391018 Ki = 45 nM T20331 CWAM95 57391019 Ki = 240 nM T20331 CG0J1A 57391020 Ki = 159 nM T20331 CHM95K 57392790 Ki = 38 nM T20331 CBSR75 57392791 Ki = 75 nM T20331 CIU0Q7 57392815 Ki = 170 nM T20331 CD31TX 57392816 Ki = 110 nM T20331 C1HN4G 57394524 Ki = 170 nM T20331 C1BNG3 57394537 Ki = 530 nM T20331 C81YWI 57396265 Ki = 3.7 nM T20331 CK8D1V 57396287 Ki = 740 nM T20331 CRP79L 57396288 Ki = 250 nM T20331 C29JBH 57396289 Ki = 360 nM T20331 C6VNM8 57398068 Ki = 34 nM T20331 C3E7AX 57398069 Ki = 290 nM T20331 C17JLA 57398070 Ki = 5000 nM T20331 C3AC5O 57398081 Ki = 49 nM T20331 CF5C9X 57398082 Ki = 80 nM T20331 CG21NR 57398083 Ki = 4300 nM T20331 CN9ED6 57398084 Ki = 2700 nM T20331 CK41BJ 57398085 Ki = 3.4 nM T20331 CEC1R9 57399726 Ki = 1851 nM T20331 CFJ7Y1 57399727 Ki = 2 nM T20331 C9SIV3 57399737 Ki = 150 nM T20331 CC72IF 57403234 Ki = 515 nM T20331 C0WY5P 57403235 Ki = 60 nM T20331 CCP7E9 57403258 Ki = 1122 nM T20331 CN9L4K 57404430 Ki = 0.9 nM T20331 CJA3K6 66677782 Ki = 5 nM T20331 C48LDN 70681100 Ki = 4 nM T20331 CQ3B1W 70681101 Ki = 0.9 nM T20331 C0B9PO 70681111 Ki = 0.8 nM T20331 CYPG86 70681118 Ki = 301 nM T20331 C81ZSO 70683225 Ki = 0.9 nM T20331 C05QUB 70683238 Ki = 8 nM T20331 CJ8WR1 70683239 Ki = 2.4 nM T20331 CG5S1X 70683240 Ki = 82 nM T20331 CAC5O7 70685314 Ki = 3.5 nM T20331 C6MW9J 70685315 Ki = 1 nM T20331 CZ4J6F 70685316 Ki = 1.2 nM T20331 C32MFH 70685339 Ki = 0.7 nM T20331 C4N5VM 70685340 Ki = 188 nM T20331 C1E5UD 70687454 Ki = 0.9 nM T20331 CKD1J6 70687455 Ki = 2.2 nM T20331 CG9Y5X 70687456 Ki = 8.9 nM T20331 CWT96B 70687457 Ki = 2 nM T20331 CST56M 70687474 Ki = 11 nM T20331 CI93CZ 70689509 Ki = 5.6 nM T20331 CHG1L3 70689510 Ki = 12 nM T20331 CID9C2 70689521 Ki = 10 nM T20331 C0CL4K 70691635 Ki = 1.7 nM T20331 C71GCS 70693713 Ki = 10 nM T20331 CW63XZ 70693714 Ki = 1.5 nM T20331 CV08YA 70693715 Ki = 1.1 nM T20331 C2R4FQ 70693716 Ki = 1.8 nM T20331 C9NRX6 70693717 Ki = 1.5 nM T20331 C96ZWB 70695681 Ki = 16 nM T20331 CT61HF 70695856 Ki = 849 nM T20331 C72PLV 70695857 Ki = 4.6 nM T20331 CGDK58 70695858 Ki = 2330 nM T20331 CE96MI 71450852 IC50 = 202 nM T20331 C32HPN 71461713 Ki = 74 nM T20331 C8QO1W 71719108 Ki > 5000 nM T20331 C9UH7J 72205287 Ki > 5000 nM T20331 CH2VP3 72205486 Ki > 5000 nM T20331 CA26US 72205877 Ki > 5000 nM T20331 CFV1X0 72711815 Ki > 1000 nM T20331 CE6KV1 72712030 Ki > 1000 nM T20331 C1X2AR 73346549 Ki > 5000 nM T20331 CPXJ28 73349570 Ki > 5000 nM T20331 C0NM1P 73351119 Ki > 1000 nM T20331 CRC73X 73354075 Ki > 1000 nM T20331 CRL10F 73354088 Ki > 5000 nM T20331 CIFL82 73354092 Ki > 5000 nM T20331 C9XCU8 73354094 Ki > 5000 nM T20331 CO26NJ 73355617 Ki > 5000 nM T20331 CUM6D5 73357147 Ki > 1000 nM T20331 CE26RI 76310949 Ki = 9 nM T20331 CN1ZR3 76321859 Ki = 10 nM T20331 CTE16Y 76321860 Ki = 41 nM T20331 CQJ70F 76325491 Ki = 4 nM T20331 CN5H4E 76329031 Ki > 10000 nM T20331 CN7ZJ3 76332712 Ki = 3 nM T20331 C95FOG 76332713 Ki = 7 nM T20331 CB3FG4 85472343 Ki = 2100 nM T20331 CW2BG8 127029975 Ki = 280 nM T20331 C7Q2WP 127030359 Ki = 220 nM T20331 CK0A1M 127031281 Ki = 140 nM T20331 C0XR6M 127041306 Ki > 10000 nM T20331 C5PA2G 127041908 Ki > 10000 nM T20331 C7TM1Y 127042243 Ki > 10000 nM T20331 C62JIE 127042244 Ki > 10000 nM T20331 C58ZTD 135430853 IC50 = 39 nM T20331 CY6T4X 135543802 IC50 = 1 nM T20331 C5WIK8 136000663 Ki = 600 nM T20331 CN4DV6 136000675 Ki = 630 nM T20331 CR52GW 136000676 Ki = 11 nM T20331 C5PEH1 136000677 Ki = 3.8 nM T20331 C7M9JL 136000678 Ki = 5 nM T20331 C4NQO8 136058109 IC50 = 54 nM T20331 C9F5MA 136058111 IC50 = 35 nM T20331 CPK6B9 136058112 IC50 = 57 nM T20331 CBI2E1 136088969 Ki = 4.3 nM T20331 CO8NB7 136088970 Ki = 3.4 nM T20331 C1K7OF 136088971 Ki = 7.4 nM T20331 C8ZAN2 145979152 Ki = 1.259 nM T20331 C4SB9P 145979291 EC50 = 790 nM T20331 CQ78WY 145979469 Ki = 1000 nM T20331 CO1M3D 145979616 Ki = 630 nM T20331 C3OXL9 145979975 Ki = 50 nM T20331 C4H9BZ 145980763 EC50 = 7.9 nM T20331 CH5MZ8 145980782 Ki = 125.89 nM T20331 CI5F7E 145980802 Ki = 1258.93 nM T20331 CP4RI5 145980997 Ki = 1.585 nM T20331 CW80EN 145981168 Ki = 5000 nM T20331 CTF1C6 145981319 Ki = 250 nM T20331 COB75I 145981742 EC50 = 500 nM T20331 C60AUT 145981829 EC50 = 790 nM T20331 COF9U8 145982156 Ki = 39.81 nM T20331 CXE2K1 145984150 Ki = 79 nM T20331 CM4VG2 145984378 Ki = 0.63 nM T20331 CG74XB 145985156 Ki = 1000 nM T20331 C5XL9U 145985176 EC50 = 5 nM T20331 C63DRI 145985639 Ki = 5000 nM T20331 C5UDH2 145986414 Ki = 199.53 nM T20331 CLEQ40 145986472 Ki = 3.162 nM T20331 CZ68SU 145986539 Ki = 3162.28 nM T20331 CGB4Y3 145987289 Ki = 1258.93 nM T20331 CI1XY0 145987577 Ki = 790 nM T20331 C4T5IJ 145987618 Ki = 1258.93 nM T20331 CL2I3Y 145987802 Ki = 1000 nM T20331 CIZ94Y 145988210 Ki = 3.981 nM T20331 CRW15D 145989250 Ki = 199.53 nM T20331 C5O8AZ 145989327 EC50 = 158.49 nM T20331 CG63IW 145989789 Ki = 31.62 nM T20331 CF5OV2 145990257 Ki = 790 nM T20331 CH50MF 145991293 EC50 = 50 nM T20331 CDX86E 145991438 Ki = 158.49 nM T20331 C6PS8F 145991876 Ki = 100 nM T20331 C7K8CT 145992181 Ki = 0.3981 nM T20331 CC72HP 145992661 Ki = 0.63 nM T20331 C5KF0O 145992989 Ki = 398.11 nM T20331 CQH29C 145993358 Ki = 15.85 nM T20331 C9Z4PM 145993376 Ki = 100 nM T20331 CAZ6I7 145993698 Ki = 25 nM T20331 CPD7M9 145994220 EC50 = 398.11 nM T20331 CQF01J 155524657 Ki = 1500 nM T20331 CCK32B 155543070 Ki = 710 nM T20331 CCZ09U 155547323 Ki = 460 nM T20331 C1T7DH 155549336 Ki = 400 nM T20331 CDT81L 155553742 Ki = 550 nM T20331 CX43VE 155561277 Ki > 10000 nM T20331 C4M9NL 155561620 Ki = 220 nM T20331 D01HFL 22054806 IC50 = 54 nM T20331 D07XFL 10007341 IC50 = 16 nM T20331 D0K0KR 9895867 IC50 = 2.7 nM T20331 D0K3QL 10030142 IC50 = 0.54 nM T20331 D0L9OS 9889267 IC50 = 53 nM T20331 D0N6HL 10052173 IC50 = 0.7 nM T20331 D0Q2IU 44439563 Ki > 1000 nM T98945 CSM4Q6 262935 Ki = 376000 nM T98945 COFC54 5347695 Ki = 11800 nM T98945 C0FJG2 5916478 Ki = 273000 nM T98945 C62WJS 6332610 Ki = 44000 nM T98945 CP3QT1 9560223 Ki = 1470 nM T98945 C9QW6K 9568045 Ki > 500000 nM T98945 C7XL2M 9573034 Ki = 1840 nM T98945 C25WST 9573756 Ki = 17300 nM T98945 CMKZ82 9574209 Ki = 4780 nM T98945 CGT32J 9994348 Ki = 1820 nM T98945 CED36V 10009347 Ki = 6400 nM T98945 C16CXQ 10033400 Ki = 900 nM T98945 CJ5CA8 10105958 Ki = 11500 nM T98945 C8OC6J 10212767 Ki = 990 nM T98945 C4C5AF 10219094 Ki = 420 nM T98945 C75TFE 10259947 Ki = 1900 nM T98945 CC46LA 10485685 Ki = 190 nM T98945 CBUF92 11228390 Ki = 1.7 nM T98945 CUIM84 11628682 Ki = 169 nM T98945 CZ78TN 11650945 Ki = 114 nM T98945 CFHX82 11837140 IC50 > 50000 nM T98945 C3RV5A 16043267 Ki = 6 nM T98945 CK7Y2E 16757513 Ki = 23 nM T98945 CL2K9U 20333093 IC50 > 50000 nM T98945 C2T4QJ 25195678 Ki = 138 nM T98945 CW1A4N 25196726 IC50 > 50000 nM T98945 C2FU9P 42618077 IC50 > 50000 nM T98945 CWXJ06 44156975 IC50 > 50000 nM T98945 C58KSV 44156976 IC50 > 50000 nM T98945 C4EZF0 44352560 Ki = 240 nM T98945 CK5HB4 44352627 Ki = 350 nM T98945 CK9BD0 44352629 Ki = 5.1 nM T98945 C0CFN6 44352635 Ki = 3.4 nM T98945 C97MNE 44352636 Ki = 7.5 nM T98945 CY4OG7 44352637 Ki = 370 nM T98945 C58IZU 44352651 Ki = 26 nM T98945 C4Z7EM 44352695 Ki = 330 nM T98945 CT3Q5N 44584806 Ki = 67 nM T98945 C5A9HE 44584807 Ki > 100 nM T98945 CJ0X2K 44584808 Ki > 100 nM T98945 CK73GW 44584809 Ki > 100 nM T98945 CI81BN 44584810 Ki > 100 nM T98945 C41POU 44584811 Ki > 100 nM T98945 C61OSN 44584812 Ki = 57 nM T98945 CB6Y4T 44584813 Ki > 100 nM T98945 CG1L4I 44584814 Ki > 100 nM T98945 CR0S1A 44584815 Ki > 100 nM T98945 CW4DN7 44584816 Ki > 100 nM T98945 CLW5C3 44584817 Ki > 100 nM T98945 CSB8X3 44584818 Ki > 100 nM T98945 CCTP19 44584819 Ki > 100 nM T98945 C29EYG 44584820 Ki > 100 nM T98945 CFR2M3 44584821 Ki > 100 nM T98945 CKG1U6 44584822 Ki > 100 nM T98945 C62FAQ 44584823 Ki > 100 nM T98945 C2K8OA 44584824 Ki > 100 nM T98945 CUF8E5 44584825 Ki > 100 nM T98945 C0X4KU 44584826 Ki > 100 nM T98945 COE8L9 44584827 Ki > 100 nM T98945 CG0KU3 44584828 Ki > 100 nM T98945 CY3V8P 44584829 Ki > 100 nM T98945 CD6ZC5 44584830 Ki > 100 nM T98945 C9UN5P 44584831 Ki > 100 nM T98945 CA0DC8 44584832 Ki > 100 nM T98945 CS27KE 44584833 Ki > 100 nM T98945 CFN4J7 44584834 Ki > 100 nM T98945 C65LUD 44584835 Ki > 100 nM T98945 CUX56H 44584836 Ki > 100 nM T98945 CS98BC 44584837 Ki > 100 nM T98945 C27ROJ 44584838 Ki > 100 nM T98945 CIB62U 44584839 Ki > 100 nM T98945 CBWC20 44584840 Ki > 100 nM T98945 CRQK05 44584841 Ki > 100 nM T98945 CT37IE 44584842 Ki > 100 nM T98945 CPL2H1 44584843 Ki > 100 nM T98945 CM29XN 44584844 Ki = 80 nM T98945 C32LWT 44584845 Ki > 100 nM T98945 CUS16Z 44584846 Ki = 30 nM T98945 CB5F0T 44584847 Ki > 100 nM T98945 CD58FL 44584848 Ki = 38 nM T98945 C3PN7C 44584849 Ki = 59 nM T98945 CQE24W 44584850 Ki > 100 nM T98945 CUQ9K4 44584863 Ki > 100 nM T98945 CE3MW2 44584948 Ki > 100 nM T98945 CQH8U7 44584950 Ki = 45 nM T98945 CPYT15 44584951 Ki = 47 nM T98945 CUZ71D 44584952 Ki = 56 nM T98945 CP2J8X 44584953 Ki = 33 nM T98945 CJKB12 44584954 Ki > 100 nM T98945 CF3Y6V 44584955 Ki > 100 nM T98945 C73YFH 44584956 Ki > 100 nM T98945 CMD1Z7 44584957 Ki > 100 nM T98945 CAOR08 44584958 Ki = 65 nM T98945 CF2LH5 44584959 Ki = 81 nM T98945 CBX8K0 44584960 Ki = 34 nM T98945 C10KCB 44584961 Ki = 38 nM T98945 C1S6KQ 44584962 Ki = 47 nM T98945 CDCH27 44584964 Ki > 100 nM T98945 C31PGM 44584965 Ki > 100 nM T98945 CQOC14 44584966 Ki > 100 nM T98945 C0GF2Q 44584967 Ki > 100 nM T98945 CF7KY4 44584968 Ki > 100 nM T98945 C4LHQ9 44584969 Ki > 100 nM T98945 C9X3FD 44584970 Ki > 100 nM T98945 CQSO90 44584971 Ki > 100 nM T98945 CD37QK 44584972 Ki > 100 nM T98945 C0G3MD 44584973 Ki > 100 nM T98945 CJM03L 44584974 Ki > 100 nM T98945 CT47PD 44584975 Ki > 100 nM T98945 CJ1P5B 44584976 Ki > 100 nM T98945 CEMD30 44584977 Ki > 100 nM T98945 CD71WT 44584978 Ki > 100 nM T98945 CG2KE0 44584979 Ki > 100 nM T98945 CLC8K5 44584980 Ki > 100 nM T98945 CF9RK1 44584981 Ki > 100 nM T98945 C9CEO7 44584982 Ki > 100 nM T98945 CXNK25 44584983 Ki > 100 nM T98945 CNA4O5 44584984 Ki > 100 nM T98945 C1J0LO 44584985 Ki > 100 nM T98945 C67DIC 44584986 Ki > 100 nM T98945 CX79JW 44584987 Ki > 100 nM T98945 CKM6J1 44584988 Ki > 100 nM T98945 C9OX8T 44584989 Ki > 100 nM T98945 CQP51O 44584990 Ki > 100 nM T98945 CP7KN4 44584991 Ki > 100 nM T98945 CJXP53 44584992 Ki > 100 nM T98945 CEB46O 44584993 Ki > 100 nM T98945 CNC7Y0 44584994 Ki > 100 nM T98945 CS02PI 44584995 Ki > 100 nM T98945 CB2K4M 44584996 Ki > 100 nM T98945 C3FE4S 44584997 Ki > 100 nM T98945 C8MAW2 44584998 Ki > 100 nM T98945 CNB4L3 44584999 Ki > 100 nM T98945 CXL76H 44585000 Ki > 100 nM T98945 C47OBC 44585001 Ki > 100 nM T98945 C3JYM7 44585002 Ki > 100 nM T98945 CG71FH 44585004 Ki > 100 nM T98945 C4CSQ2 44585005 Ki > 100 nM T98945 C7ZO5P 44585006 Ki > 100 nM T98945 CK5VW7 44585007 Ki > 100 nM T98945 CG0OR5 44585008 Ki > 100 nM T98945 C78MRO 44585009 Ki > 100 nM T98945 CR27AE 44585010 Ki > 100 nM T98945 C8M7DI 44585011 Ki > 100 nM T98945 COEC52 44585012 Ki > 100 nM T98945 CKG8S2 44585013 Ki > 100 nM T98945 CST23K 44585014 Ki > 100 nM T98945 C4BSZ6 44585015 Ki > 100 nM T98945 CO1E8Z 44585016 Ki > 100 nM T98945 C5KJ9Q 44585017 Ki > 100 nM T98945 CQX41M 44585018 Ki > 100 nM T98945 CI6AW8 44585019 Ki > 100 nM T98945 C34MRQ 44585020 Ki > 100 nM T98945 CNQR65 44585021 Ki > 100 nM T98945 C8Z4WQ 44585022 Ki > 100 nM T98945 CWEI08 44585023 Ki > 100 nM T98945 C1UF2C 44585024 Ki > 100 nM T98945 C32TRO 44585025 Ki > 100 nM T98945 CU9CH7 44585026 Ki > 100 nM T98945 C5WVR1 44585027 Ki > 100 nM T98945 CC4P1B 44585028 Ki > 100 nM T98945 C4ZQP1 44585029 Ki > 100 nM T98945 CGML74 44585030 Ki > 100 nM T98945 C8SM9K 44585031 Ki > 100 nM T98945 CWC2Y9 44585032 Ki > 100 nM T98945 CZH7M3 44585033 Ki > 100 nM T98945 CZ7S2E 44585034 Ki > 100 nM T98945 CG60WN 44585035 Ki > 100 nM T98945 CMV32T 44585036 Ki > 100 nM T98945 CN74EF 44585037 Ki > 100 nM T98945 CCTM89 44585038 Ki > 100 nM T98945 CC25VQ 44585039 Ki > 100 nM T98945 CY3CG4 44585040 Ki > 100 nM T98945 CV1F3G 44585041 Ki > 100 nM T98945 C8KOE2 44585042 Ki > 100 nM T98945 CG9CO3 44585043 Ki > 100 nM T98945 CZ9F8X 44585044 Ki = 115 nM T98945 CC8MJ0 44585045 Ki = 48 nM T98945 C9MR4W 44585046 Ki > 100 nM T98945 CB7N5J 44585047 Ki > 100 nM T98945 CH7C1E 44585048 Ki > 100 nM T98945 CG0UK7 44585049 Ki = 103 nM T98945 C7PYW8 44585050 Ki > 100 nM T98945 C5JHS4 44585051 Ki = 58 nM T98945 C1PDB6 44585052 Ki > 100 nM T98945 CL9PD0 44585053 Ki > 100 nM T98945 CC0V7O 44585054 Ki > 100 nM T98945 C8UBS3 44585055 Ki > 100 nM T98945 CA1PS3 44585056 Ki = 50 nM T98945 CE2PV8 44585057 Ki > 100 nM T98945 CBM2Y7 44585058 Ki > 100 nM T98945 CZVN12 44585059 Ki > 100 nM T98945 C7T3LQ 44585060 Ki > 100 nM T98945 CKH27O 44585061 Ki > 100 nM T98945 CAZ34N 44585062 Ki = 93 nM T98945 C4VD2W 44585063 Ki > 100 nM T98945 CQV2W1 44585064 Ki > 100 nM T98945 C3YJL1 44585065 Ki > 100 nM T98945 CGA7K6 44585066 Ki > 100 nM T98945 CLBV32 44585067 Ki > 100 nM T98945 CQIJ72 44585068 Ki > 100 nM T98945 CG02SN 44585069 Ki > 100 nM T98945 C98HFK 44585070 Ki > 100 nM T98945 C9T5CZ 44585071 Ki > 100 nM T98945 CRL9H6 44585072 Ki > 100 nM T98945 CHA0M1 44585073 Ki > 100 nM T98945 C1F3XD 44585074 Ki > 100 nM T98945 C82EPA 44585075 Ki > 100 nM T98945 CGX5C2 44585076 Ki > 100 nM T98945 CF8B5L 44585077 Ki > 100 nM T98945 CP7K4R 44585078 Ki > 100 nM T98945 CT2MV6 44585079 Ki > 100 nM T98945 C1R9XI 44585080 Ki > 100 nM T98945 CXC08A 44585081 Ki > 100 nM T98945 CLC7S0 44585082 Ki > 100 nM T98945 C0QH7B 44585083 Ki > 100 nM T98945 CX70KM 44585084 Ki > 100 nM T98945 CO0N2T 44585085 Ki > 100 nM T98945 C42TGS 44585086 Ki > 100 nM T98945 C58ZDW 44585087 Ki > 100 nM T98945 C45NBG 44585088 Ki > 100 nM T98945 CVD73E 44585089 Ki > 100 nM T98945 C49VDL 44585090 Ki > 100 nM T98945 CC61AT 44585091 Ki > 100 nM T98945 C2F8QP 44585092 Ki > 100 nM T98945 CIP31K 44585093 Ki > 100 nM T98945 COJ28W 44585094 Ki > 100 nM T98945 C9RGX0 44585095 Ki > 100 nM T98945 C4ZUP3 44585096 Ki > 100 nM T98945 C06VHK 44585097 Ki > 100 nM T98945 CPJ9K4 44585099 Ki > 100 nM T98945 CWT6A4 44585100 Ki > 100 nM T98945 C9MWI6 44585101 Ki > 100 nM T98945 CNZ81Q 44585102 Ki = 39 nM T98945 CE4WN9 44585107 Ki = 42 nM T98945 C6X1HU 44585113 Ki > 100 nM T98945 C8X1KW 44585114 Ki > 100 nM T98945 CU5KY2 44585115 Ki > 100 nM T98945 CU27NO 44585116 Ki > 100 nM T98945 CGK50M 44585117 Ki > 100 nM T98945 CQD4Z8 44585118 Ki > 100 nM T98945 C94ZCT 44585119 Ki = 57 nM T98945 C2ZWE4 44585120 Ki > 100 nM T98945 CK7XM0 44585121 Ki > 100 nM T98945 CN3AD9 44585122 Ki > 100 nM T98945 C7RI5O 44585123 Ki > 100 nM T98945 C0ZBN3 44585124 Ki > 100 nM T98945 CC75XO 44585125 Ki > 100 nM T98945 CWNB15 44585126 Ki > 100 nM T98945 C57HGE 44585127 Ki = 80 nM T98945 CI09DY 44585128 Ki > 100 nM T98945 CJ7LF5 44585129 Ki = 30 nM T98945 CO93HF 44585130 Ki = 38 nM T98945 C0MJN2 44585131 Ki > 100 nM T98945 C8V5GT 44585132 Ki = 59 nM T98945 CIRV70 44585133 Ki > 100 nM T98945 C2RNK5 44585134 Ki > 100 nM T98945 CRW3B9 44585135 Ki > 100 nM T98945 CVTE96 44585136 Ki = 53 nM T98945 C2W5AH 44585137 Ki = 45 nM T98945 C9TFD6 44585138 Ki = 47 nM T98945 C7X2UH 44585139 Ki = 56 nM T98945 C1H2WG 44585140 Ki > 100 nM T98945 CRL0A6 44585141 Ki > 100 nM T98945 CT1N4A 44585142 Ki > 100 nM T98945 CZ6SO5 44585143 Ki > 100 nM T98945 CG8R2Y 44585144 Ki = 65 nM T98945 CS4TQ6 44585145 Ki = 81 nM T98945 CO56MF 44585146 Ki > 100 nM T98945 C9SW4V 44585147 Ki > 100 nM T98945 C46BYS 44585148 Ki > 100 nM T98945 CIJ0Z8 44585149 Ki > 100 nM T98945 C79UBQ 44585150 Ki > 100 nM T98945 C8YO5T 44585151 Ki > 100 nM T98945 CW5A2K 44585152 Ki > 100 nM T98945 C56DTX 44585153 Ki > 100 nM T98945 CFDC58 44585154 Ki > 100 nM T98945 CVL28O 44585155 Ki > 100 nM T98945 C6C4MS 44585156 Ki > 100 nM T98945 C4C7HG 44585157 Ki > 100 nM T98945 CDI21X 44585158 Ki > 100 nM T98945 CKIJ08 44585159 Ki > 100 nM T98945 C8R5YX 44585160 Ki > 100 nM T98945 CYC8R9 44585161 Ki > 100 nM T98945 CCRD92 44585162 Ki > 100 nM T98945 CJV7X2 44585163 Ki > 100 nM T98945 C5TDU2 44585164 Ki > 100 nM T98945 CQFC87 44585165 Ki > 100 nM T98945 CUA85D 44593129 Ki = 89 nM T98945 C7P8EK 44593130 Ki = 404 nM T98945 C4JS9X 44593146 Ki = 22 nM T98945 CQ4OK8 44593147 Ki = 69 nM T98945 C20JPC 44593148 Ki = 12 nM T98945 CUZ62D 44593168 Ki = 42 nM T98945 C6S5JH 44593169 Ki = 46 nM T98945 CNT7J8 44593170 Ki = 423 nM T98945 C0Q9CE 44593171 Ki = 812 nM T98945 CWP01R 44593172 Ki = 1768 nM T98945 CV07SM 44593173 Ki = 100000 nM T98945 CEW2O5 44593174 Ki = 100000 nM T98945 CB80ER 44593175 Ki = 100000 nM T98945 CE3CR0 44593197 Ki = 100000 nM T98945 C2YPS6 44593198 Ki = 100000 nM T98945 C7P5LR 44593199 Ki = 100000 nM T98945 CN3EB5 44612015 Ki = 800 nM T98945 CGF70P 45486343 Ki = 3020 nM T98945 CNOP07 45486344 Ki = 63 nM T98945 C4G3BC 45486345 Ki = 7490 nM T98945 CJ73BT 45486346 Ki = 78 nM T98945 CF9I7Y 45486347 Ki = 553 nM T98945 C1NIR6 45486348 Ki = 1070 nM T98945 CAJQ48 45486349 Ki = 627 nM T98945 C6EB3A 45486350 Ki = 1430 nM T98945 CW8RA2 45486351 Ki = 1320 nM T98945 CQS4W0 45486352 Ki = 2730 nM T98945 CSX01I 45486353 Ki = 9710 nM T98945 C9ETC4 45486354 Ki = 53 nM T98945 CVPG40 45486356 Ki = 1.6 nM T98945 CSQ2K4 45486357 Ki = 1 nM T98945 CL4D9S 45486358 Ki = 3.3 nM T98945 CDE58N 46191000 Ki = 285 nM T98945 CAJL68 46191001 Ki = 702 nM T98945 CG1HV0 46191002 Ki = 1.5 nM T98945 C8FP5E 46191072 Ki = 7340 nM T98945 C7NM3V 46191073 Ki = 37 nM T98945 C3X0OE 46191074 Ki = 24 nM T98945 CWL5Q8 46191148 Ki = 6 nM T98945 C5YX7K 46191149 Ki = 3 nM T98945 C8Z6SQ 46191150 Ki = 3.7 nM T98945 CYN8K9 46191291 Ki = 40 nM T98945 C9NC7I 46191292 Ki = 19 nM T98945 C2INC9 46191293 Ki = 3 nM T98945 CR7I8G 46191363 Ki = 3.6 nM T98945 CV1X4F 46191364 Ki = 1.4 nM T98945 CT26LP 46191365 Ki = 0.84 nM T98945 CQGL01 46191433 Ki = 12 nM T98945 CQ1MA3 46191434 Ki = 6.3 nM T98945 C32SJP 46191435 Ki = 23 nM T98945 C97QIZ 46191505 Ki = 405 nM T98945 CJZA45 46232267 IC50 > 50000 nM T98945 C3PLE6 46232269 IC50 > 50000 nM T98945 C3U8HV 46232270 IC50 > 50000 nM T98945 CYA73D 46232312 IC50 > 50000 nM T98945 C9Q7YX 53317374 Ki = 27900 nM T98945 CA86OS 53317375 Ki = 1130 nM T98945 C93QWB 53318957 Ki = 5610 nM T98945 C4W1DB 53320248 Ki = 1130 nM T98945 CLO86W 53321180 Ki = 580 nM T98945 CGZC91 53321290 Ki = 173000 nM T98945 C7QEI1 53321291 Ki = 460 nM T98945 CFOI53 53322612 Ki = 1550 nM T98945 CWA7B3 53323948 Ki = 1040 nM T98945 CSYV84 53325117 Ki = 1940 nM T98945 CQ7D3S 53325118 Ki = 1350 nM T98945 CO6TG4 53325236 Ki = 1420 nM T98945 CO0R2M 53325237 Ki = 1200 nM T98945 C8G4SM 53326426 Ki = 1460 nM T98945 CSP13L 53380708 Ki = 0.83 nM T98945 C2NYC4 53380709 Ki = 1.9 nM T98945 CB2W7R 56660089 Ki = 13 nM T98945 CTN23H 56660090 Ki = 1110 nM T98945 CCG0B8 56660091 Ki = 2390 nM T98945 CD1X9B 56663556 Ki = 3200 nM T98945 C9P3SV 56667001 Ki = 5.9 nM T98945 C6K5AI 56670442 Ki = 970 nM T98945 CX3F7D 56673930 Ki = 102 nM T98945 CVA9L6 56673931 Ki = 238 nM T98945 CY28PE 56673932 Ki = 1385 nM T98945 C2GXS8 56677267 Ki = 9.7 nM T98945 CEPU28 56680566 Ki = 142 nM T98945 CV3H4S 56683904 Ki = 6.3 nM T98945 C8ON3V 70684173 Ki = 3020 nM T98945 C4O8IR 70684174 Ki = 7490 nM T98945 CF78WO 70684175 Ki = 1070 nM T98945 CU9BW3 70684182 Ki = 2730 nM T98945 CGX63U 70684183 Ki = 3500 nM T98945 CYK60H 70686317 Ki = 1 nM T98945 C0TCG9 70686318 Ki = 3.3 nM T98945 C2XUM9 70686319 Ki = 3400 nM T98945 C4ESI6 70688429 Ki = 1.6 nM T98945 C87OHL 70690464 Ki = 63 nM T98945 C3R9EA 70690465 Ki = 78 nM T98945 C2MD9T 70690466 Ki = 1320 nM T98945 CUCP34 70690475 Ki = 53 nM T98945 CA9YT3 70692619 Ki = 1430 nM T98945 C9MVW4 70694663 Ki = 553 nM T98945 C41VFE 70694672 Ki = 9710 nM T98945 CDEV58 70694673 Ki = 0.81 nM T98945 CG4C9F 70696704 Ki = 627 nM T98945 C6TO1L 71450124 Ki = 1000 nM T98945 C8F5YQ 71451941 Ki > 1000 nM T98945 CGD6J4 71451942 Ki = 400 nM T98945 CY86ZW 71453763 Ki = 1300 nM T98945 C5I3EB 71453792 Ki = 500 nM T98945 CT51YJ 71453793 Ki = 1.4 nM T98945 C7WM6Z 71455497 Ki = 430 nM T98945 C35YRK 71457282 Ki = 2600 nM T98945 C2YEU4 71457318 Ki = 760 nM T98945 CB9MG1 71459125 Ki = 12.4 nM T98945 C0N8UR 71460934 Ki = 2.9 nM T98945 CDLP98 71460935 Ki = 5.3 nM T98945 CIS3R0 71460936 Ki = 4100 nM T98945 CK1X0W 71462644 Ki = 9 nM T98945 CGR35S 71462645 Ki = 1200 nM T98945 CQNG13 71608634 Ki = 9.8 nM T98945 C6HAL4 73345659 Ki > 100 nM T98945 CK7O6Q 73350255 Ki = 53 nM T98945 C4APW2 75593416 Ki = 680 nM T98945 CJ2W9V 75593418 Ki = 27 nM T98945 C29QOJ 76310654 Ki = 980 nM T98945 CAT6S5 76310655 Ki = 9550 nM T98945 CG87ZE 76310656 Ki = 7300 nM T98945 CQ7TE3 76310980 Ki = 8 nM T98945 CV8Z5G 76314290 Ki = 800 nM T98945 CULA07 76314608 Ki = 89 nM T98945 C6BT0I 76314609 Ki = 6 nM T98945 C6ZXN7 76314610 Ki = 1.9 nM T98945 CGB4J9 76317836 Ki = 650 nM T98945 C7G4XB 76317837 Ki = 560 nM T98945 CFXK67 76317855 Ki = 950 nM T98945 C6JAY9 76318181 Ki = 123 nM T98945 CYJ1I9 76318182 Ki = 21 nM T98945 CH3N0A 76321557 Ki = 1980 nM T98945 CF78UP 76321572 Ki = 1070 nM T98945 CX5I2O 76321887 Ki = 18 nM T98945 CA5K8R 76321888 Ki = 591 nM T98945 CMYK97 76325157 Ki = 980 nM T98945 CZ62KS 76328735 Ki = 2300 nM T98945 C4LG2O 76328736 Ki = 2100 nM T98945 C2J7OP 76329062 Ki = 25 nM T98945 CDC1J5 76329063 Ki = 33 nM T98945 CIY15Q 76332398 Ki = 2550 nM T98945 CL2ZX3 76332418 Ki = 2800 nM T98945 CX2VL4 76336024 Ki = 1120 nM T98945 CGZN04 76336044 Ki = 11000 nM T98945 C0ET8W 137630787 Ki = 1 nM T98945 CC3V7S 137631353 Ki = 3 nM T98945 C2JV6R 137631479 Ki = 0.4 nM T98945 C53MJF 137631755 Ki = 3 nM T98945 CN26ME 137631991 Ki = 11.7 nM T98945 CUOC87 137632800 Ki = 2 nM T98945 C5VFZ9 137633317 Ki = 3.1 nM T98945 C73DJB 137633620 Ki = 5 nM T98945 CBNJ52 137633770 Ki = 5.9 nM T98945 CRN21S 137633930 Ki = 50 nM T98945 CP8DN5 137634404 Ki = 0.9 nM T98945 CAIC85 137634503 Ki = 3 nM T98945 C0T3NR 137635077 Ki = 5 nM T98945 C9MUE6 137636542 Ki = 4.5 nM T98945 CG95RB 137636600 Ki = 4 nM T98945 C4GHK8 137636619 Ki = 4 nM T98945 CG5Q8T 137636730 Ki = 1.7 nM T98945 CH8AU1 137636950 Ki = 13 nM T98945 CDVJ93 137637528 Ki = 18 nM T98945 C5DX1A 137637600 Ki = 2.3 nM T98945 CDY46K 137637620 Ki = 260 nM T98945 C87STU 137638937 Ki = 30 nM T98945 C5L0NC 137639050 Ki = 4 nM T98945 CBH65X 137639397 Ki = 12 nM T98945 CN0FY7 137639688 Ki = 0.5 nM T98945 CJMG20 137640300 Ki = 13 nM T98945 CB2Z9N 137640311 Ki = 4 nM T98945 CERC30 137640559 Ki = 1.8 nM T98945 C35AYG 137641095 Ki = 3 nM T98945 CUM15D 137641134 Ki = 140 nM T98945 CQ76RK 137641874 Ki = 6 nM T98945 CO3S8F 137641997 Ki = 6 nM T98945 CMA50S 137642172 Ki = 0.5 nM T98945 C5AM0F 137642389 Ki = 5 nM T98945 CNC1O3 137642533 Ki = 36 nM T98945 CA5PJ2 137642642 Ki = 2.6 nM T98945 CX53VG 137642650 Ki = 38 nM T98945 CHI60U 137642806 Ki = 0.7 nM T98945 C7W9US 137643496 Ki = 1.1 nM T98945 C7PR9K 137644391 Ki = 1.5 nM T98945 C98VOE 137645351 Ki = 1.5 nM T98945 C0NWD3 137645581 Ki = 15 nM T98945 CQ6SI9 137645677 Ki = 7 nM T98945 CJT5C4 137646929 Ki = 4 nM T98945 C8WED4 137647032 Ki = 0.9 nM T98945 C76BDY 137647768 Ki = 8 nM T98945 CD3CZ6 137647834 Ki = 3 nM T98945 C64QUK 137648887 Ki = 50 nM T98945 CBP37G 137649385 Ki = 7 nM T98945 C2N9LT 137650514 Ki = 6 nM T98945 COR8J3 137652054 Ki = 27 nM T98945 CJX57S 137652059 Ki = 4 nM T98945 CVC56D 137652453 Ki = 11 nM T98945 CUP70F 137652558 Ki = 3.4 nM T98945 CJVG81 137652912 Ki = 23 nM T98945 CPO80U 137653066 Ki = 5 nM T98945 CN5VC7 137653379 Ki = 8.1 nM T98945 C34XTZ 137653755 Ki = 2 nM T98945 CUHM58 137653788 Ki = 3 nM T98945 C4B8DK 137654788 Ki = 9 nM T98945 C4XTJ7 137655341 Ki = 1.4 nM T98945 C7W1GU 137655527 Ki = 4 nM T98945 CBRA14 137655621 Ki = 4.7 nM T98945 CI78BN 137656445 Ki = 3 nM T98945 CD9N0S 137656589 Ki = 8 nM T98945 CV7T5U 137656624 Ki = 16.7 nM T98945 CI3A4J 137657514 Ki = 1.1 nM T98945 CO09SX 137658594 Ki = 3 nM T98945 CZY51S 137659359 Ki = 0.6 nM T98945 C8J2FS 137659865 Ki = 1 nM T98945 CXYA13 137660373 Ki = 2.4 nM T98945 C37WVK 137660935 Ki = 18 nM T98945 CGBP12 137661234 Ki = 3.1 nM T98945 CSI79D 137661408 Ki = 4 nM T98945 CV3NU9 137661582 Ki = 4.8 nM T98945 CDP9F6 145979561 Ki = 41 nM T98945 C0FVL7 145980400 Ki = 825 nM T98945 C7U6AC 145980921 Ki = 60 nM T98945 C1PY3D 145982564 Ki = 2600 nM T98945 C0F2HS 145982570 Ki = 290 nM T98945 C9BAM3 145982642 Ki = 2500 nM T98945 CO1L7J 145982755 Ki = 260 nM T98945 CH49CQ 145982874 Ki = 700 nM T98945 CL4F2V 145983062 Ki = 74 nM T98945 C8P4IY 145983083 Ki = 280 nM T98945 CD4V6Y 145983456 Ki = 100 nM T98945 C0VPE7 145983531 Ki = 990 nM T98945 CMN3C0 145983800 Ki = 210 nM T98945 CKY29N 145984016 Ki = 140 nM T98945 C71KAW 145984052 Ki = 140 nM T98945 C7Y5TR 145984180 Ki = 330 nM T98945 CI2E5Y 145984243 Ki = 74 nM T98945 CP4M8O 145984298 Ki = 130 nM T98945 CR0E5D 145984449 Ki = 130 nM T98945 CBK18Y 145984711 Ki = 110 nM T98945 C9W1TO 145984728 Ki = 80 nM T98945 CZ9MK3 145984956 Ki = 990 nM T98945 C6VYO5 145985131 Ki = 500 nM T98945 C0DJ8X 145985285 Ki = 170 nM T98945 CME81P 145985674 Ki = 3000 nM T98945 CMT30D 145985833 Ki = 64 nM T98945 CN96XK 145985989 Ki = 200 nM T98945 C6UA9H 145986239 Ki = 190 nM T98945 CG7LW4 145987687 Ki = 38 nM T98945 C3C2LW 145989654 Ki = 614 nM T98945 C4IW1B 145989737 Ki = 240 nM T98945 C4ACG5 145990382 Ki = 600 nM T98945 CZJY41 145990864 Ki = 21.5 nM T98945 CB9FH7 145992096 Ki = 250 nM T98945 C9KC4Q 145993075 Ki = 60 nM T98945 D05JJL 44584947 Ki = 23 nM T98945 D0A6FZ 75593419 Ki = 4.3 nM T98945 D0Y9PH 45486355 Ki = 0.81 nM T30082 D04AIT 5280445 Ki = 65800 nM T30082 D04QLR 3180 IC50 = 181 nM T30082 D05QNO 2968 IC50 = 1000 nM T30082 D06OMW 3052776 IC50 = 19 nM T30082 D06XWB 854026 IC50 = 33 nM T30082 D07HBX 338 IC50 = 346000 nM T30082 D07HOB 60838 Ki = 50.5 nM T30082 D07MGA 72281 IC50 = 2476100 nM T30082 D07XYV 54766 IC50 = 30000 nM T30082 D08SKH 4114 IC50 = 760 nM T30082 D08USJ 4456 IC50 = 2400 nM T30082 D08VYV 4168 IC50 > 20000 nM T30082 D09MWJ 2092 IC50 = 18 nM T30082 D09QDP 4380 IC50 > 500000 nM T30082 D09QEI 4740 IC50 = 6600 nM T30082 D0B3HD 2519 IC50 = 7250 nM T30082 D0E6YQ 1935 IC50 = 7.53 nM T30082 D0K8KX 5280343 Ki = 38300 nM T30082 D0L4JT 5333 IC50 = 145240 nM T30082 D0NJ3V 4680 IC50 = 24330 nM T30082 D0NS6H 3152 IC50 = 2 nM T30082 D0O2WB 4991 IC50 = 360 nM T30082 D0Q0RC 3290 IC50 = 260 nM T30082 D0R0MW 5329102 IC50 = 5870 nM T30082 D0R1QE 3672 IC50 = 235110 nM T30082 D0R9VR 9651 Ki = 61.9 nM T30082 D0S2UG 26757 IC50 > 500000 nM T30082 D0TR5X 3386 IC50 = 130 nM T30082 D0U5SI 4913 IC50 = 1000 nM T30082 D0UU9Y 4938 IC50 = 6400 nM T30082 D0W8SJ 4199 IC50 = 85000 nM T30082 D0W8WB 2353 IC50 = 100 nM T30082 D0WY5Q 77991 IC50 = 54 nM T30082 D0X7DE 4449 IC50 = 1037 nM T30082 D00VUI 6199 IC50 = 6480 nM T30082 D01LYX 65872 IC50 = 5 nM T30082 D02EVF 6112 IC50 = 1 nM T30082 D07CIN 192706 IC50 = 21 nM T30082 D07SDQ 969516 IC50 > 5000 nM T30082 D0B1FE 3194 IC50 = 6200 nM T30082 D0B6IZ 137905 Ki > 100000 nM T30082 D0C3UC 208907 IC50 = 52400 nM T30082 D0L9QM 59568713 IC50 = 9940 nM T30082 D0M3IN 1188 IC50 = 9000 nM T30082 D0T5AW 442894 IC50 = 3720 nM T30082 D0U3EP 445154 IC50 > 5000 nM T30082 D0G9HY 118717433 IC50 = 96.3 nM T30082 D0I7KU 118717425 IC50 = 91.8 nM T30082 D0RN2X 442126 IC50 = 390000 nM T30082 D02UOE 160142 Ki > 100000 nM T30082 D09JVV 5983 IC50 = 0.008 ug.mL-1 T30082 D09PTA 132228 IC50 = 148 nM T30082 D0AM8W 198752 IC50 < 500 nM T30082 D0B2BQ 135462830 IC50 = 0.33 nM T30082 D0F1VQ 60811 IC50 = 92.9 nM T30082 D0L8QQ 3655 IC50 = 164 nM T30082 D0S1VV 119053 Ki = 2090 nM T30082 C4F9OB 342 IC50 = 45.71 nM T30082 CXU4W0 650 Ki > 100000 nM T30082 CT6RA0 2317 IC50 = 7244.36 nM T30082 C6HD1N 2879 IC50 = 1.82 nM T30082 CKHG70 3017 IC50 = 1900 nM T30082 CQ6GW7 3039 IC50 = 627 nM T30082 C0RFA2 3102 Ki > 100000 nM T30082 CFS16G 3450 Ki = 37000 nM T30082 CUQ05A 3564 IC50 = 23700 nM T30082 C7VMZ3 4108 IC50 = 5370.32 nM T30082 C37AQO 4970 IC50 > 100000 nM T30082 C93BJO 5039 IC50 = 650 nM T30082 C8F5QC 5077 IC50 = 35200 nM T30082 CYZL84 5579 IC50 = 191866.87 nM T30082 C8GZO5 5741 IC50 = 20 nM T30082 CKB56J 5824 IC50 = 42.1 nM T30082 CNL74P 6760 IC50 = 8.6 ug.mL-1 T30082 C4IU5T 6889 Ki > 100000 nM T30082 C5NIV3 7088 IC50 = 7400 nM T30082 C5EUF4 7108 IC50 = 7300 nM T30082 CY1BV2 7237 IC50 = 10 nM T30082 C3RKS6 7241 IC50 = 4900 nM T30082 CLE8Y0 7422 IC50 = 3.981 nM T30082 C0CR3O 7473 IC50 = 100 nM T30082 CA70BO 7530 IC50 = 218.78 nM T30082 CK4PA0 7731 IC50 = 3630.78 nM T30082 C0A5JC 7809 IC50 = 4900 nM T30082 C1WR2I 7813 IC50 = 36.31 nM T30082 C37NWX 7929 IC50 = 4900 nM T30082 C6NQ4X 8246 IC50 = 0.043 nM T30082 CJL02I 8307 Ki = 200 nM T30082 C1ER4M 9336 Ki = 1.63 nM T30082 CCQ42B 9603 IC50 = 9.55 nM T30082 C9T7HX 9606 IC50 = 1 nM T30082 CTY1W5 9820 Ki = 10 nM T30082 C25CYL 10434 Ki > 100000 nM T30082 C47FYB 10662 Ki > 100000 nM T30082 C2G5AW 11066 IC50 > 100000 nM T30082 CZP3G7 11100 Ki > 100000 nM T30082 COGY52 11321 Ki > 100000 nM T30082 C7U0TW 11747 Ki > 100000 nM T30082 C53FYO 11840 Ki > 100000 nM T30082 CKR3L9 12116 Ki > 100000 nM T30082 CU5KZ0 13005 Ki > 100000 nM T30082 CJ2GH1 13006 Ki > 100000 nM T30082 C3E4AQ 13837 IC50 = 2387811.28 nM T30082 CG1LI5 14313 Ki > 100000 nM T30082 C2XQ4P 15384 IC50 = 972.75 nM T30082 CPXJ40 17233 IC50 = 229086.77 nM T30082 C4FW7E 18475 Ki > 100000 nM T30082 CON67V 19853 IC50 = 5500 nM T30082 CTE5Z9 22006 IC50 = 39 nM T30082 C0M1GZ 22486 IC50 = 1129795.91 nM T30082 C03DVR 22519 IC50 = 1000000 nM T30082 CDS1J0 26007 IC50 = 847227.41 nM T30082 C7S3JO 26257 Ki > 100000 nM T30082 CV59WB 28535 IC50 = 3013.01 nM T30082 C38JQX 31261 Ki > 100000 nM T30082 C3ZUD9 37851 IC50 = 439541.62 nM T30082 CN8A2G 38296 Ki > 100000 nM T30082 C7HE8W 38333 Ki > 100000 nM T30082 C0VK3I 39834 Ki > 100000 nM T30082 CVS6A8 40634 IC50 = 186400 nM T30082 C2NY3T 40710 IC50 = 597035.29 nM T30082 C8Z6TM 43402 Ki > 100000 nM T30082 CB3MZ8 46612 IC50 = 3111.72 nM T30082 C46RKB 46780 IC50 > 10000 nM T30082 CM94KL 47020 IC50 = 1875 nM T30082 CY1LU4 48688 IC50 = 2824.88 nM T30082 CQJ24R 51298 IC50 > 10000 nM T30082 CUNJ73 61209 Ki > 100000 nM T30082 C6U7FB 62539 Ki > 100000 nM T30082 C1NQ8E 65188 IC50 = 150000 nM T30082 C09AHX 68081 IC50 = 69000 nM T30082 CEKW96 68115 Ki > 100000 nM T30082 CL5B7Z 68119 Ki > 100000 nM T30082 CT70IY 68126 IC50 = 4900 nM T30082 C54XNY 68261 IC50 = 62500 nM T30082 C27NHT 69147 Ki > 100000 nM T30082 CN0ID1 69282 Ki > 100000 nM T30082 CW54JA 69288 Ki > 100000 nM T30082 C6BEN0 70945 Ki > 100000 nM T30082 CR6Z7K 72119 IC50 = 100000 nM T30082 C5KW4H 72311 Ki = 320 nM T30082 CTY16O 73191 IC50 = 68000 nM T30082 C2I7WP 74721 IC50 = 1700 nM T30082 CV8R4B 76561 Ki > 100000 nM T30082 CVJ78Y 79690 Ki > 100000 nM T30082 CF8DH5 80661 IC50 = 1158777.36 nM T30082 CY7N0S 80922 IC50 = 4900 nM T30082 CAPG58 87502 Ki > 100000 nM T30082 C0EH3Z 88695 Ki > 100000 nM T30082 CE6M5B 89121 IC50 = 49730 nM T30082 CN16GW 91420 IC50 = 84722.74 nM T30082 C70KGR 92036 Ki > 100000 nM T30082 C13IQL 93772 Ki > 100000 nM T30082 CCP9A2 95069 IC50 > 50000 nM T30082 C8YU9Z 95415 Ki > 100000 nM T30082 CH91PI 95447 Ki > 100000 nM T30082 C0RTJ6 100313 IC50 = 1940 nM T30082 CAET12 101464 Ki = 89300 nM T30082 CR3E9L 103786 Ki > 100000 nM T30082 C0QSW4 104849 IC50 = 25118.86 nM T30082 CTV6F8 107935 IC50 = 126700 nM T30082 C4K3TN 114909 IC50 = 127180 nM T30082 C7KJ3B 114917 IC50 > 50000 nM T30082 CLF2C0 115097 IC50 = 360 nM T30082 C7WZK3 120734 IC50 > 100000 nM T30082 CVB9H1 121587 IC50 = 3200 nM T30082 CVH8G6 122824 Ki = 24700 nM T30082 CJV02W 124069 IC50 > 100000 nM T30082 CN3OE7 132619 IC50 = 1.2 nM T30082 C20LIY 136371 Ki > 100000 nM T30082 CTU83D 137777 Ki > 100000 nM T30082 CHAN02 138508 Ki > 100000 nM T30082 CYX5V0 142278 Ki > 100000 nM T30082 CZ1IF9 148724 IC50 > 100 ug.mL-1 T30082 CCF76B 151146 IC50 = 87902.25 nM T30082 CF3I2J 156793 IC50 = 121600 nM T30082 C5X1YU 160254 Ki = 6410 nM T30082 CVT05J 160306 IC50 = 6.8 nM T30082 CS8RE2 160512 IC50 = 191100 nM T30082 CNMW72 160522 IC50 > 100000 nM T30082 C84VQZ 160875 IC50 > 100000 nM T30082 CJT1U2 163001 IC50 = 1840 nM T30082 C4IRY2 164676 Ki > 100000 nM T30082 C28RAT 165208 IC50 = 28000 nM T30082 C1EAJ8 172972 IC50 = 0.33 nM T30082 CR7KU8 179849 IC50 = 1610 nM T30082 CC92WL 179850 IC50 = 476 nM T30082 CMS7P5 189686 IC50 > 100000 nM T30082 CX54PW 192442 IC50 = 6.761 nM T30082 C3SGD8 196830 IC50 = 28.84 nM T30082 C73HEY 203361 IC50 = 505000 nM T30082 C1UW4K 204303 IC50 = 1770000 nM T30082 CT8KV4 205772 IC50 = 56 nM T30082 CH2AJ6 216347 IC50 = 38 nM T30082 CVMD70 218049 IC50 = 1000000 nM T30082 C6W8MB 219592 Ki > 100000 nM T30082 COQ09W 219605 Ki > 100000 nM T30082 C25BHS 222475 Ki > 100000 nM T30082 CN35KE 222570 Ki > 100000 nM T30082 CP4W3S 229680 Ki > 100000 nM T30082 C0NGE1 231178 IC50 = 81.28 nM T30082 CARJ43 231563 IC50 = 10000 nM T30082 CW5N2U 232124 Ki = 1500 nM T30082 C0KV5M 236566 Ki > 100000 nM T30082 CE6U1D 237515 Ki > 100000 nM T30082 C92OSL 241331 Ki > 100000 nM T30082 COU8X4 249262 IC50 = 380 nM T30082 C7X5SP 249597 IC50 = 620 nM T30082 C4N8IF 252525 IC50 > 30000 nM T30082 CN75IX 255296 IC50 = 22000 nM T30082 C5Y6QK 261619 IC50 > 100000 nM T30082 CHP1J7 262695 Ki > 100000 nM T30082 CDL3E1 262696 Ki > 100000 nM T30082 C6PU5E 270291 IC50 = 59200 nM T30082 CBV0N9 275005 Ki > 100000 nM T30082 CF62QN 275182 IC50 > 100000 nM T30082 C06INE 275192 IC50 = 10730 nM T30082 C4HQ7V 284016 IC50 > 100000 nM T30082 C08WNV 317405 IC50 > 100000 nM T30082 CY3C1Q 323438 IC50 = 51000 nM T30082 CU35JW 324062 IC50 = 1310 nM T30082 CNP1J9 334704 IC50 = 67000 nM T30082 C5EI4Q 354120 IC50 = 131170 nM T30082 CHL04T 362574 IC50 > 100000 nM T30082 CKS3U9 366710 Ki > 100000 nM T30082 CSR38O 367141 IC50 = 28000 nM T30082 C5V0SH 386338 IC50 = 7300 nM T30082 C54EGJ 402658 IC50 = 38200 nM T30082 C9E5NG 402660 IC50 = 2980 nM T30082 CGKY63 402662 IC50 = 9100 nM T30082 CDCN80 402664 IC50 = 391100 nM T30082 C34VZP 402665 IC50 = 68800 nM T30082 C98AUK 402666 IC50 = 166100 nM T30082 C7HME8 439246 IC50 = 2045000 nM T30082 C18OIX 441064 IC50 = 97000 nM T30082 CW4NS2 441251 IC50 = 9900 nM T30082 CK8SE3 441593 IC50 = 452000 nM T30082 CRN10Y 442113 IC50 = 27 nM T30082 CYI84X 442127 IC50 = 28000 nM T30082 CK3H2X 442638 IC50 = 93000 nM T30082 C0KUP1 442979 IC50 = 39810.72 nM T30082 CP26JX 443685 IC50 > 200000 nM T30082 CC0JT1 443689 IC50 = 187630 nM T30082 CPGB82 443722 IC50 = 100 nM T30082 C4M9PZ 443723 IC50 = 20070 nM T30082 C6X5KE 443725 IC50 = 3870 nM T30082 CV6Z1N 443739 IC50 = 1430 nM T30082 CK4V7H 453077 IC50 = 11480 nM T30082 CYMH94 471008 IC50 = 21840 nM T30082 CMO53J 475411 IC50 = 16270 nM T30082 C3AYB0 479059 IC50 > 100000 nM T30082 C74VWI 480865 IC50 = 15500 nM T30082 CGU9L8 511106 IC50 > 100000 nM T30082 CT0P5D 511111 IC50 > 100000 nM T30082 CN67CR 555078 IC50 > 100000 nM T30082 CL2CH5 559371 IC50 = 8750 nM T30082 CTWM69 586418 Ki > 100000 nM T30082 CH1E7N 590628 Ki > 100000 nM T30082 CCJQ96 599378 Ki > 100000 nM T30082 C0SXA3 604519 IC50 = 658 nM T30082 CL5E6W 607775 IC50 > 10000 nM T30082 CC61DL 609857 IC50 = 36.31 nM T30082 C1QE9B 612726 IC50 = 335 nM T30082 CQ94TR 639465 IC50 = 7200 nM T30082 C3JLN7 642384 IC50 = 1260 nM T30082 CC9J6K 652654 IC50 = 409200 nM T30082 CV8GA2 657093 IC50 = 89 nM T30082 C9MC2E 657348 IC50 = 28 nM T30082 CK5V3P 667498 IC50 = 9890 nM T30082 CR1E5K 667801 IC50 = 6200 nM T30082 C7R8DL 675624 IC50 > 100000 nM T30082 C3DPV8 705751 Ki = 1450000 nM T30082 CA2LD8 738882 IC50 > 200000 nM T30082 CTL9W3 741894 IC50 = 500 nM T30082 CC3PD7 748096 IC50 > 200000 nM T30082 C50NVY 784043 IC50 = 1200 nM T30082 C4TAX6 784405 IC50 = 850 nM T30082 CXEL98 789450 IC50 = 41 nM T30082 C5PDK8 802516 IC50 = 18710 nM T30082 CMB76R 805935 IC50 > 200000 nM T30082 CB3GD4 818016 Ki = 59800 nM T30082 CQL19V 822847 IC50 = 318 nM T30082 C1QUN8 823959 IC50 = 1150 nM T30082 CRT9N1 826073 IC50 > 100 ug.mL-1 T30082 CU2MK8 828189 IC50 = 8128.31 nM T30082 C29EOV 830741 IC50 = 9900 nM T30082 C6WT1U 840737 IC50 > 200000 nM T30082 C3XY5A 882744 IC50 = 3390 nM T30082 C28RCY 886888 IC50 > 200000 nM T30082 C4AM0D 887037 IC50 = 140000 nM T30082 C6QO9M 895655 IC50 = 120000 nM T30082 CM06JU 906525 IC50 > 100000 nM T30082 C5BR8V 908164 IC50 > 100000 nM T30082 C6LP2A 924755 IC50 > 100000 nM T30082 C3S6JC 972870 IC50 = 12000 nM T30082 CL8T1M 973113 IC50 > 200000 nM T30082 CXBQ97 1086746 IC50 = 458 nM T30082 CJ8H6A 1131663 IC50 = 43000 nM T30082 CFE1M2 1131698 IC50 > 200000 nM T30082 C9HG2Y 1207322 IC50 = 78.9 nM T30082 CRP1I7 1211924 IC50 > 100000 nM T30082 CED67Q 1237217 IC50 = 6300 nM T30082 CGV7M9 1245748 IC50 = 90000 nM T30082 CR1J2F 1375660 IC50 > 200000 nM T30082 CX9N6W 1376254 IC50 > 200000 nM T30082 C8ENO6 1395053 IC50 = 30 nM T30082 CO0K8X 1549992 IC50 < 10 ug.mL-1 T30082 CIK9V0 1593398 IC50 = 1.4 nM T30082 CWTV42 1713189 Ki > 100000 nM T30082 C0EX9G 1755771 Ki > 100000 nM T30082 CX3C0J 1761244 IC50 = 5000 nM T30082 CB0ZP3 1812008 Ki > 100000 nM T30082 C3FQD8 1906162 Ki > 100000 nM T30082 CV3TR1 1943896 IC50 > 1000000 nM T30082 C3O6MN 1972026 Ki > 100000 nM T30082 CI6ZU8 2133593 IC50 > 100000 nM T30082 CF37ZA 2147394 Ki > 100000 nM T30082 CESV82 2258987 IC50 = 5100 nM T30082 CJD8B3 2305233 Ki > 100000 nM T30082 CN4U9J 2359994 IC50 = 5900 nM T30082 CC5J8U 2723754 Ki = 101 nM T30082 COQ45C 2723878 Ki = 6300 nM T30082 C09FTW 2728676 IC50 = 4100 nM T30082 C0OZQ2 2731126 Ki > 100000 nM T30082 CNKV06 2731127 Ki > 100000 nM T30082 CEM2C8 2731732 Ki > 100000 nM T30082 C2HOC5 2731733 Ki > 100000 nM T30082 CVC36I 2731902 Ki > 100000 nM T30082 CG62CN 2731904 Ki > 100000 nM T30082 C8JAT4 2733068 IC50 = 1300 nM T30082 CVD82J 2734800 Ki > 100000 nM T30082 CZ2TV6 2739707 IC50 = 2600 nM T30082 C76YPA 2741467 Ki = 2870 nM T30082 CBEC45 2742082 IC50 > 15000 nM T30082 CN3KA4 2743222 IC50 = 100 nM T30082 C4MAI9 2747679 IC50 = 15000 nM T30082 C9R5LQ 2749125 Ki > 100000 nM T30082 C84DSN 2749126 Ki > 100000 nM T30082 CT6JX7 2776817 IC50 = 16000 nM T30082 C8HE5U 2777804 IC50 = 14000 nM T30082 C84VWR 2784639 Ki > 100000 nM T30082 CDCB42 2786143 Ki > 100000 nM T30082 CV4YZ2 2796017 Ki = 263.15 nM T30082 CE3S2O 2796640 IC50 = 8000 nM T30082 CFU21P 2797788 IC50 = 389000 nM T30082 C2H3AG 2802899 Ki = 61.4 nM T30082 C65GYK 2810357 Ki = 241.14 nM T30082 CU6OI3 2810689 Ki = 54.84 nM T30082 CM8HT1 2811064 Ki = 21.29 nM T30082 COBU39 2813142 Ki = 47.34 nM T30082 CYV1U9 2814953 Ki = 95.3 nM T30082 CD4JI6 2822603 Ki = 22.78 nM T30082 C0UKM1 2825872 IC50 = 27000 nM T30082 C8K9UF 2878002 IC50 = 448000 nM T30082 CQD5I9 2911244 IC50 = 31000 nM T30082 C1XFI4 2970848 IC50 = 120000 nM T30082 CTU27I 2981783 IC50 > 1000000 nM T30082 CRQ94D 2999234 IC50 > 100000 nM T30082 CRU43A 3000083 IC50 = 45000 nM T30082 C1BM9V 3001811 IC50 = 22310 nM T30082 CC4OL6 3004425 IC50 = 5248.07 nM T30082 CLN03H 3026641 IC50 = 1510080.15 nM T30082 C9QOY1 3029941 Ki = 16300 nM T30082 CNYW30 3036637 IC50 = 1540000 nM T30082 CF3A1Q 3038398 IC50 = 176 nM T30082 CZVE24 3041340 IC50 = 63000 nM T30082 C0JO2G 3055247 IC50 = 290 nM T30082 CVN73X 3071771 IC50 = 28 nM T30082 CS5ET2 3071772 IC50 = 330 nM T30082 CG09EQ 3071773 IC50 = 210 nM T30082 CP2Y7N 3071774 IC50 = 900 nM T30082 CZ6BA1 3071775 IC50 = 740 nM T30082 C9M5PQ 3071776 IC50 = 610 nM T30082 CI9VN7 3071777 IC50 = 470 nM T30082 CC6W7T 3071778 IC50 = 460 nM T30082 CIKF06 3071779 IC50 = 260 nM T30082 CL2HU7 3071780 IC50 = 180 nM T30082 CR4GK9 3072018 IC50 = 12487 nM T30082 CM0S9H 3072029 IC50 = 381 nM T30082 C4P5ZF 3072030 IC50 = 208 nM T30082 CC9S8H 3072501 IC50 = 200 nM T30082 CBLG95 3072502 IC50 = 120 nM T30082 CS3L6G 3072503 IC50 = 650 nM T30082 CIW2K3 3072504 IC50 = 83 nM T30082 C2KN6J 3072505 IC50 = 160 nM T30082 CEU74K 3072506 IC50 = 260 nM T30082 CC56GR 3072507 IC50 = 520 nM T30082 C4PCM1 3072508 IC50 = 370 nM T30082 CHD8L0 3072509 IC50 = 310 nM T30082 CU61MK 3072510 IC50 = 690 nM T30082 CS1I6C 3072512 IC50 = 440 nM T30082 CU20TQ 3072513 IC50 = 640 nM T30082 C3KTC4 3072514 IC50 = 680 nM T30082 C6QM9J 3072515 IC50 = 630 nM T30082 CXLH39 3072518 IC50 = 1300 nM T30082 CI87YF 3073076 Ki = 9.333 nM T30082 CQ8FC6 3074014 IC50 = 80 nM T30082 C2WZG6 3074016 IC50 = 40 nM T30082 CO7N8L 3074341 IC50 = 125 nM T30082 CO6NL8 3074344 IC50 = 133 nM T30082 C09SID 3075610 IC50 = 350 nM T30082 C1OGL8 3075611 IC50 = 460 nM T30082 COW6E8 3075612 IC50 = 100 nM T30082 CK2FX6 3077650 IC50 = 9300 nM T30082 CJ0LY2 3077884 IC50 = 162.18 nM T30082 CU9Z2X 3083559 IC50 = 5600 nM T30082 CN5Z4H 3084319 IC50 = 21 nM T30082 C3EY8Z 3087084 IC50 = 12.5 nM T30082 C9OL5T 3087086 IC50 = 4.2 nM T30082 CHEA42 3088389 IC50 = 500 nM T30082 C3UE8V 3088445 IC50 = 27000 nM T30082 C6RT2B 3088563 IC50 = 5400 nM T30082 C1AM0S 3114312 Ki > 100000 nM T30082 C61RSW 3126152 Ki > 100000 nM T30082 CCP07Y 3264931 Ki > 100000 nM T30082 CB21VL 3321360 Ki > 100000 nM T30082 CZV6G2 3329233 Ki > 100000 nM T30082 CH32KQ 3353663 IC50 = 220 nM T30082 C6NH9P 3469206 Ki > 100000 nM T30082 C3BT1N 3478673 IC50 = 5800 nM T30082 C10GCK 3527426 Ki > 100000 nM T30082 C3T1CV 3531512 Ki > 100000 nM T30082 CXE3M5 3537759 Ki = 6430 nM T30082 COY89G 3738100 IC50 = 3850 nM T30082 C5UM2D 3821945 Ki = 3280 nM T30082 C7KWS6 3966943 IC50 = 5.3 nM T30082 CB49EF 3988576 IC50 = 18380 nM T30082 CU17BR 4088910 Ki > 100000 nM T30082 CCBK12 4246119 IC50 < 100000 nM T30082 CC1GF9 4338240 Ki > 100000 nM T30082 C8KV7I 4350924 Ki > 100000 nM T30082 CPX4V3 4352680 IC50 = 89.13 nM T30082 C0V6QI 4369935 Ki > 100000 nM T30082 C42FGN 4384851 Ki > 100000 nM T30082 CJ16WI 4385120 IC50 = 534564.36 nM T30082 CN9C3V 4513067 Ki > 100000 nM T30082 CF2GX1 4551826 IC50 = 135.1 nM T30082 C5IZS9 4636426 IC50 > 1000 nM T30082 CBIY84 4655388 IC50 = 2500 nM T30082 CE6ZA4 4720373 IC50 > 500000 nM T30082 CAOH69 4789430 IC50 = 4000 nM T30082 CK9AT5 4792504 IC50 = 2400 nM T30082 CDV3O6 4846969 Ki = 100 nM T30082 C9MY1I 4885038 IC50 = 8320 nM T30082 C5NJ3A 5004413 Ki > 100000 nM T30082 CNMY06 5038499 Ki > 100000 nM T30082 CL69XS 5127299 IC50 = 425 nM T30082 C7A0CD 5152006 IC50 = 7850 nM T30082 C5B4MJ 5251958 IC50 = 141253.75 nM T30082 C0D3PO 5281671 Ki = 3100 nM T30082 C0L6SF 5281846 IC50 > 100 ug.mL-1 T30082 C5LGJ1 5282362 IC50 > 500000 nM T30082 CY9RO7 5315699 IC50 > 200000 nM T30082 COB0W2 5316525 IC50 = 2400000 nM T30082 CN4V2F 5320438 IC50 > 250000 nM T30082 C2OF8J 5324562 IC50 = 180000 nM T30082 CM98QZ 5351364 IC50 = 17680 nM T30082 C5U2EK 5351434 IC50 = 22040 nM T30082 C8HQN1 5376026 IC50 > 10000 nM T30082 C9LSB5 5462442 EC50 = 19 nM T30082 C1Y0UG 5468622 IC50 = 80000 nM T30082 C67WRC 5469427 IC50 = 15120 nM T30082 C57CAV 5471832 IC50 = 70000 nM T30082 CMI50J 5471833 IC50 > 100000 nM T30082 C3KW9E 5471834 IC50 = 6000 nM T30082 C5RE8A 5471835 IC50 = 50000 nM T30082 CO0R1W 5471836 IC50 = 70000 nM T30082 CH6DT9 5481958 Ki = 3100 nM T30082 CC6IV0 5481968 Ki = 3100 nM T30082 CH8AJ6 5481969 Ki = 3100 nM T30082 CMOI48 5481973 Ki = 3100 nM T30082 CLD04R 5488283 IC50 = 12 nM T30082 CP69QB 5702326 IC50 = 1600 nM T30082 C81LVR 5702328 IC50 = 4400 nM T30082 CP46OW 5713121 IC50 = 500 nM T30082 C8M0OD 5716903 IC50 = 91500 nM T30082 CLE17J 5743439 IC50 = 628058.36 nM T30082 CGHW32 5747382 IC50 = 76 nM T30082 C9L6KZ 5919802 IC50 = 7630 nM T30082 CR67NI 6333010 IC50 = 2111 nM T30082 CK2MJ6 6333011 IC50 = 2604 nM T30082 C8SZQ4 6410685 IC50 = 470 nM T30082 C58FPO 6410811 IC50 = 260000 nM T30082 CF5CI3 6410821 IC50 = 34000 nM T30082 CLPR37 6420076 IC50 = 3660 nM T30082 CYJ4I8 6476665 IC50 > 100000 nM T30082 C2LS0C 6479236 IC50 = 99900 nM T30082 CIL06S 6486743 IC50 = 8000 nM T30082 CNB34I 6540271 Ki = 27.9 nM T30082 C20VIR 6603845 IC50 = 9887 nM T30082 C6EFT0 6712920 IC50 = 0.43 nM T30082 CZD7R6 6884840 IC50 = 88500 nM T30082 CY4GC1 6918635 IC50 = 101 nM T30082 CNE62Z 6918662 IC50 = 812.83 nM T30082 CAV73I 7065962 IC50 = 192 nM T30082 CQG5N3 7098687 IC50 > 100000 nM T30082 C7BZ0N 7945979 IC50 > 5000 nM T30082 C7NTA9 8618826 IC50 = 14000 nM T30082 CGOY14 8618834 IC50 = 46000 nM T30082 C8KM7A 9405885 IC50 = 57000 nM T30082 C1BEW3 9406020 IC50 = 115000 nM T30082 C3B5QD 9578246 IC50 = 45 nM T30082 C4MO0B 9583618 IC50 = 6700 nM T30082 C1A6JL 9583695 Ki = 2070 nM T30082 CQ4Z1X 9583696 Ki = 521.34 nM T30082 CI0W6F 9583697 Ki = 2350 nM T30082 CPM0Y2 9625548 IC50 = 81100 nM T30082 C5M3KG 9638193 IC50 = 81400 nM T30082 C8XKM7 9794806 IC50 = 5 nM T30082 C9TZ6S 9798502 IC50 = 8.299 nM T30082 C80OXI 9804733 IC50 = 6 nM T30082 CS0W6A 9816573 IC50 = 1850 nM T30082 CBIF14 9818098 IC50 = 47000 nM T30082 CU2XN7 9819233 IC50 = 13 nM T30082 CFHP83 9822470 IC50 = 175 nM T30082 CVDM07 9828345 IC50 = 0.6 nM T30082 CNA7Q2 9836764 Ki = 54.95 nM T30082 CKMO29 9838394 IC50 = 0.29 ug.mL-1 T30082 CG6W8R 9839754 IC50 = 750 nM T30082 CJ63BD 9843116 IC50 = 82.5 nM T30082 CQV42M 9844067 IC50 = 3.631 nM T30082 CM0BX3 9850331 IC50 = 0.7 nM T30082 CKA8W7 9851127 IC50 = 0.3 nM T30082 C84EYV 9856666 IC50 = 15500 nM T30082 C5TKP4 9859434 IC50 = 5 nM T30082 C4VHS5 9859456 IC50 = 676.08 nM T30082 C6N2KV 9860965 IC50 = 400 nM T30082 C02WVA 9862743 IC50 > 3000 nM T30082 CZ1O9A 9863613 IC50 = 58 nM T30082 CF05ZV 9864626 IC50 = 760 nM T30082 C2S1ZR 9866271 IC50 > 3000 nM T30082 C2NLZ5 9886877 IC50 = 88 nM T30082 C1FSQ3 9887137 IC50 = 350 nM T30082 C26MUN 9887376 IC50 = 9.772 nM T30082 CM1CP9 9888147 IC50 = 15 nM T30082 CME5I4 9894056 IC50 = 0.07 nM T30082 CF1H2S 9901561 IC50 = 208.93 nM T30082 C7K6OX 9904798 IC50 = 1640 nM T30082 C94UJV 9905831 IC50 = 22 nM T30082 CH2RN9 9909244 Ki = 0.7943 nM T30082 CY3FW6 9924349 IC50 = 13.3 nM T30082 CE8M7Y 9928503 Ki = 620 nM T30082 C8EM1X 9945661 Ki = 19.95 nM T30082 C6F3YB 9949561 Ki = 7.762 nM T30082 COH8P4 9949799 IC50 > 3000 nM T30082 C2EF4O 9951444 IC50 > 3000 nM T30082 CE69LQ 9952812 IC50 = 6500 nM T30082 CFW16Y 9958700 IC50 > 30000 nM T30082 CYLG46 9959612 IC50 = 0.81 nM T30082 CC3G7N 9961034 IC50 = 29.3 nM T30082 CI2HX5 9969592 IC50 > 3000 nM T30082 C3DKO1 9973113 IC50 = 6800 nM T30082 C95XQY 9973416 IC50 > 50000 nM T30082 CA9X0F 9974154 IC50 = 98 nM T30082 C2KUR6 9974344 IC50 = 108 nM T30082 CP7J3X 9975443 IC50 = 65 nM T30082 CLJM18 9975444 IC50 = 205 nM T30082 CKAL79 9975916 IC50 = 54 nM T30082 CP3QN4 9976101 IC50 = 30 nM T30082 CSUQ31 9976190 IC50 = 700 nM T30082 C56KCN 9976499 IC50 = 120 nM T30082 C2WYT7 9976761 IC50 = 0.95 nM T30082 CI6T9D 9976843 IC50 = 11 nM T30082 CCV3X2 9976949 IC50 = 812 nM T30082 C9WXP0 9978621 IC50 = 1348.96 nM T30082 CH53OD 9979312 IC50 = 18 nM T30082 CFH1O0 9992823 IC50 = 56.7 nM T30082 C65OXD 9993507 IC50 = 660 nM T30082 CBFN90 9996198 IC50 = 320 nM T30082 CBM5Q2 9996767 IC50 = 218.78 nM T30082 CFG9W4 9997900 IC50 = 80 nM T30082 C3B8DU 9998815 IC50 = 11 nM T30082 CS6M2W 9998921 IC50 = 27000 nM T30082 C57ZOX 9998997 IC50 = 89 nM T30082 C2MH1Q 9999994 IC50 = 59 nM T30082 CZ74LC 10000487 IC50 = 81 nM T30082 CI47MJ 10001179 Ki = 21.88 nM T30082 CPC4B2 10001409 IC50 = 2652 nM T30082 CGYW94 10002656 IC50 = 240 nM T30082 C4LQ5E 10002693 IC50 = 590 nM T30082 C9R6BK 10003266 EC50 = 19 nM T30082 C6V8NY 10008886 IC50 = 33113.11 nM T30082 CW6C3X 10013554 IC50 = 87 nM T30082 C9TC3J 10019926 IC50 = 170 nM T30082 CI0DP1 10020679 IC50 = 5.754 nM T30082 CS60QN 10022823 IC50 = 6360 nM T30082 CAYM38 10023740 IC50 = 4.5 nM T30082 C54IKC 10024209 IC50 = 29 nM T30082 C07UOE 10027926 IC50 = 14 nM T30082 CI3D7M 10038341 IC50 = 30 nM T30082 CH0R1M 10038557 IC50 = 17000 nM T30082 CH71ZI 10039975 IC50 > 50000 nM T30082 C30ZHN 10040889 IC50 = 302 nM T30082 CF31SR 10043367 IC50 = 113 nM T30082 C2E5OH 10044206 IC50 = 23 nM T30082 C6H9RQ 10045172 IC50 = 1800 nM T30082 C17ERY 10046173 IC50 = 331 nM T30082 CI5NS7 10047821 IC50 = 390 nM T30082 CM75QS 10047824 IC50 = 100 nM T30082 C0BAO9 10050190 IC50 = 25.8 nM T30082 C5M2LI 10050814 IC50 = 180 nM T30082 CYK0F4 10060655 IC50 = 436.52 nM T30082 C1YLC4 10066130 IC50 = 2070141.35 nM T30082 CDX8M0 10066364 IC50 = 17 nM T30082 CFT8Z0 10067904 IC50 = 120 nM T30082 C6IQ8T 10069534 IC50 = 64 nM T30082 CX3ER1 10069858 IC50 = 2.8 nM T30082 CAMU42 10070183 IC50 = 333 nM T30082 C9HT2M 10073246 IC50 = 3140 nM T30082 C01TNX 10083133 IC50 = 28 nM T30082 C9C2DJ 10088398 IC50 = 52 nM T30082 C8UGH2 10088400 IC50 = 99 nM T30082 C7MZ6T 10089125 IC50 = 20 nM T30082 CE5HZ6 10089805 IC50 = 15000 nM T30082 CY6E7S 10090059 IC50 = 165.96 nM T30082 CE64DB 10090328 IC50 = 16 nM T30082 CPK57C 10090665 IC50 = 2300 nM T30082 CN52EC 10090965 IC50 = 36 nM T30082 CPWD05 10091114 IC50 = 707.95 nM T30082 CLG9Y2 10091498 IC50 = 77 nM T30082 CHW7N8 10091961 IC50 = 9 nM T30082 CVJ76F 10092326 IC50 = 50 nM T30082 C6SNP5 10093505 IC50 = 47 nM T30082 CRX29E 10093769 IC50 = 440 nM T30082 CEKX28 10094001 IC50 > 50000 nM T30082 C49HMN 10094694 IC50 = 853 nM T30082 CWD41K 10097011 IC50 = 1.4 nM T30082 CO1X6R 10097526 IC50 = 40 nM T30082 CTI26V 10098048 IC50 = 22630 nM T30082 C4FGP2 10101669 IC50 = 6000 nM T30082 CTS5E8 10104685 IC50 = 623 nM T30082 CI70JE 10109540 IC50 > 50000 nM T30082 C68RJB 10110147 IC50 = 2.8 nM T30082 CTQ95J 10110914 IC50 = 4.266 nM T30082 C8EQJ9 10112210 EC50 = 100 nM T30082 CIV15Q 10113978 IC50 = 930 nM T30082 C27MKW 10114327 IC50 > 31622.78 nM T30082 CSX92P 10126521 IC50 > 50000 nM T30082 C6L5QN 10131681 IC50 = 2300 nM T30082 C6NDV0 10132004 IC50 > 3000 nM T30082 C1B9MQ 10150601 IC50 > 50000 nM T30082 CA5J4V 10150622 IC50 > 50000 nM T30082 CO6I2N 10159339 IC50 = 33 nM T30082 C50QMS 10178169 IC50 = 9 nM T30082 C9L0IV 10198698 IC50 = 489 nM T30082 CQB9D0 10200831 IC50 = 54 nM T30082 C5MY9G 10204472 IC50 = 36.5 nM T30082 C36DNM 10215997 IC50 > 50000 nM T30082 CVFE26 10241903 IC50 = 3760 nM T30082 CU48ZN 10243146 IC50 = 158 nM T30082 CWZ5S0 10245631 IC50 = 40.8 nM T30082 CKAP27 10246305 IC50 = 9 nM T30082 CK2MC6 10247257 IC50 = 800 nM T30082 COL3W1 10247326 Ki = 7.079 nM T30082 C8K2AD 10248127 IC50 = 70 nM T30082 CL4E1T 10249516 IC50 = 1100 nM T30082 CQ6HR0 10249830 IC50 = 22 nM T30082 CHV6W1 10249992 IC50 = 64 nM T30082 CUZ5K4 10250049 IC50 = 393 nM T30082 CC86YL 10250291 IC50 = 35 nM T30082 CU6B5G 10255032 IC50 = 19498.45 nM T30082 C81ONP 10255275 IC50 = 1 nM T30082 CW23ZK 10255470 IC50 = 6 nM T30082 C9EBY2 10264399 IC50 = 15000 nM T30082 C8MAO5 10268794 Ki = 29400 nM T30082 C96ZXH 10269924 IC50 = 350 nM T30082 CB2K1F 10287897 IC50 > 50000 nM T30082 C0TWQ3 10292083 IC50 = 12 nM T30082 CO58BI 10295924 IC50 = 652 nM T30082 CV5B1A 10308583 IC50 > 50000 nM T30082 CJ0VN5 10310052 IC50 > 50000 nM T30082 CG8C9A 10314859 IC50 = 1600 nM T30082 CJ29KL 10315567 Ki = 100 nM T30082 CUK65V 10315690 IC50 = 1200 nM T30082 CF3HU9 10316494 IC50 = 140 nM T30082 CW70XT 10317424 IC50 = 22.91 nM T30082 CES2W1 10317677 IC50 = 3100 nM T30082 C7NRO3 10317909 IC50 = 12000 nM T30082 C1HK9D 10318438 IC50 = 10000 nM T30082 C7A3TZ 10320833 IC50 = 2.6 nM T30082 CEK31N 10321405 IC50 = 230 nM T30082 C3Q4JP 10335000 IC50 = 270 nM T30082 CPRK30 10337156 IC50 = 3500 nM T30082 C4J8NO 10337506 IC50 = 6000 nM T30082 CP8RT3 10337833 IC50 = 1000 nM T30082 CX3PI2 10338707 IC50 = 10 nM T30082 CMP61S 10340599 IC50 = 182 nM T30082 CTO45L 10341985 IC50 = 1330 nM T30082 CGZ5B9 10342292 Ki = 3100 nM T30082 CV3E1B 10358790 IC50 = 12000 nM T30082 CRI5E2 10360601 IC50 = 110 nM T30082 C4VY3L 10363687 IC50 = 26 nM T30082 C26CMB 10367598 IC50 = 30 nM T30082 CK6G3Z 10368032 IC50 = 1.1 nM T30082 C3H0MY 10372514 Ki = 12.2 nM T30082 C0G1JP 10379901 Ki = 20000 nM T30082 C25WON 10382902 IC50 = 2000 nM T30082 C4UN0X 10383200 IC50 = 13 nM T30082 CPY98N 10383204 IC50 = 1400 nM T30082 C4PE3K 10383261 IC50 = 830 nM T30082 C9TD6W 10384292 IC50 = 46 nM T30082 CLJK16 10385010 IC50 = 2680 nM T30082 C6YV7A 10385042 IC50 = 3000 nM T30082 C0PYS7 10385270 IC50 = 76 nM T30082 C3Z4ID 10386522 IC50 = 9400 nM T30082 CXU2T0 10387306 IC50 = 4.6 nM T30082 C2EWU3 10389859 IC50 = 340 nM T30082 CB9S7E 10400903 IC50 = 800 nM T30082 CAI1D7 10402718 IC50 = 1610 nM T30082 CDZV38 10403528 IC50 = 6100 nM T30082 CF3ME6 10404467 IC50 = 340 nM T30082 C30YGD 10405626 IC50 = 7.194 nM T30082 CK9BG4 10407316 IC50 = 13300 nM T30082 CA89CQ 10408960 IC50 = 376 nM T30082 CB2Z3Y 10410110 EC50 = 2700 nM T30082 C8E4YN 10411163 IC50 = 5.4 nM T30082 CZHX93 10411563 IC50 = 2.4 nM T30082 CC5WG8 10416369 IC50 = 26.2 nM T30082 C9G7HY 10425802 IC50 = 45 nM T30082 CB3NC2 10425948 IC50 = 86000 nM T30082 CY4I2F 10426283 IC50 = 2570.4 nM T30082 C9LKY8 10426799 IC50 = 13 nM T30082 CSI7Y6 10427747 IC50 = 1100 nM T30082 C9M4VA 10428809 IC50 = 13 nM T30082 C3AX2Y 10429940 IC50 = 125 nM T30082 C35WUQ 10431427 IC50 = 30 nM T30082 CT79BG 10431485 IC50 = 847 nM T30082 CA04FU 10433807 IC50 = 1500 nM T30082 CU12MF 10433924 IC50 = 28840.32 nM T30082 C0E6JC 10439720 IC50 = 12660 nM T30082 C0H3TC 10448720 IC50 = 43900 nM T30082 CR9L5G 10449628 IC50 = 810 nM T30082 CC75LI 10450489 IC50 = 13 nM T30082 C5X3BL 10450804 IC50 = 1200 nM T30082 C7KR3A 10451317 IC50 = 50 nM T30082 CG23NW 10451362 Ki = 8.71 nM T30082 CYD3O4 10453018 IC50 = 224 nM T30082 CI7C9Y 10464995 IC50 > 10000 nM T30082 CFN3I9 10472189 IC50 = 74710 nM T30082 CK2QA7 10473914 IC50 = 8.8 nM T30082 C60QFP 10474803 IC50 = 8 nM T30082 CU21VN 10476544 IC50 > 50000 nM T30082 C7W8EX 10478397 IC50 = 55 nM T30082 CHM50O 10481357 IC50 = 0.3 nM T30082 C7IZC8 10492974 IC50 = 1000000 nM T30082 CKD0Q6 10496874 IC50 = 4786.3 nM T30082 C2C3XA 10498282 IC50 = 47 nM T30082 C7J2KT 10502606 IC50 = 3560 nM T30082 C4QB5Z 10503812 IC50 = 2500 nM T30082 CK5W8X 10505674 IC50 = 1760 nM T30082 CY8F2J 10515621 IC50 = 22.91 nM T30082 C92OYA 10518487 IC50 = 3715.35 nM T30082 C5Y7TM 10521068 IC50 = 131 nM T30082 C4M6EH 10521536 IC50 = 11000 nM T30082 CF5E2S 10521609 Ki = 29 nM T30082 CGH7U6 10526350 IC50 = 1910 nM T30082 CAJF06 10529304 IC50 = 37 nM T30082 CWUY91 10539341 IC50 = 69400 nM T30082 CO5SV7 10539945 IC50 = 40000 nM T30082 CD9CO7 10545404 IC50 = 65000 nM T30082 C98RWG 10545891 IC50 = 161 nM T30082 C9EKA4 10548335 IC50 = 12.8 nM T30082 CM3UP4 10550262 IC50 = 3110 nM T30082 C5LEQ9 10552178 IC50 = 38 nM T30082 CSE98A 10553699 IC50 = 5.7 nM T30082 CTUJ81 10553759 IC50 = 4 nM T30082 CFR06U 10555466 IC50 = 170 nM T30082 CE93NH 10564954 IC50 = 80000 nM T30082 CJ0N1R 10569957 IC50 = 2847.5 nM T30082 CV1I8T 10571010 IC50 = 71 nM T30082 CFZ0U2 10573193 IC50 = 13.6 nM T30082 CF91YT 10573262 IC50 = 1819.7 nM T30082 CIS15A 10573780 IC50 = 245.3 nM T30082 CX0A2M 10575968 IC50 = 250 nM T30082 CB6OS5 10578606 IC50 = 31 nM T30082 C3A0CW 10587149 IC50 = 500000 nM T30082 CYSD36 10593041 IC50 = 40 nM T30082 CG09QV 10593268 IC50 = 1000 nM T30082 C3XYI4 10597848 IC50 = 11223 nM T30082 CCDQ76 10598017 IC50 = 83 nM T30082 CW9HE7 10598755 IC50 = 176 nM T30082 CVD9A1 10610498 IC50 = 1490 nM T30082 CTM40A 10615903 IC50 = 5654.5 nM T30082 CAP4U2 10617077 IC50 = 52 nM T30082 C9C1GH 10617967 IC50 = 740000 nM T30082 CQ83HS 10620599 IC50 = 243 nM T30082 C2LRS9 10622407 IC50 = 100 nM T30082 CV1PG0 10623652 IC50 = 13000 nM T30082 CY93KL 10625415 IC50 = 1.6 nM T30082 CN28TC 10638188 IC50 = 500000 nM T30082 C1VKX9 10638726 IC50 = 389.05 nM T30082 C9UKR0 10641198 IC50 = 35000 nM T30082 C3IG4V 10646592 IC50 > 100000 nM T30082 CW61PA 10647381 IC50 > 100000 nM T30082 CHZJ42 10647656 IC50 = 0.56 nM T30082 CV3S0G 10648705 IC50 = 36 nM T30082 CWE41Q 10655805 Ki > 100000 nM T30082 C97XMS 10660565 IC50 = 62000 nM T30082 CQJ31U 10662773 IC50 = 128.82 nM T30082 C01EQG 10662852 IC50 = 319 nM T30082 CZ59MX 10663695 IC50 = 285 nM T30082 CN4AM2 10672184 IC50 = 0.82 nM T30082 C1OSU0 10672185 IC50 = 28 nM T30082 CG0AC9 10682905 IC50 = 16218.1 nM T30082 C0O2KM 10683827 IC50 = 1000000 nM T30082 CA4F2Y 10687047 IC50 = 170000 nM T30082 C9V0LI 10689771 IC50 = 56000 nM T30082 CSIC19 10690207 IC50 = 2020 nM T30082 CV9R3W 10691270 IC50 = 45 nM T30082 CPC8D5 10695859 IC50 = 0.7 nM T30082 CD35YF 10711007 IC50 = 169.82 nM T30082 CNR15Z 10713570 IC50 = 740 nM T30082 CR4AM9 10716472 IC50 = 264 nM T30082 C7TES2 10720926 IC50 > 100000 nM T30082 CF19GP 10721441 IC50 = 70 nM T30082 CG4Z8N 10721720 IC50 = 13 nM T30082 CUW26T 10728025 IC50 > 10000000 nM T30082 CL1BE8 10729509 IC50 = 25000 nM T30082 CRD47N 10730136 IC50 = 2193.5 nM T30082 CZ9TD2 10730721 IC50 = 50000 nM T30082 CCF63R 10733266 IC50 = 50000 nM T30082 CIF7T8 10738642 IC50 = 180 nM T30082 CXFK03 10742628 IC50 = 13 nM T30082 CXN9A5 10743162 IC50 = 14 nM T30082 CRK9M1 10753951 IC50 = 30 nM T30082 CT68IS 10757271 IC50 = 231 nM T30082 CXVH42 10762160 Ki = 35 nM T30082 C4O5KP 10763156 IC50 = 127 nM T30082 CDAR18 10764956 IC50 = 1090 nM T30082 CB96TA 10768189 IC50 = 100 nM T30082 CO93ID 10774617 IC50 = 39810.72 nM T30082 C2AN5S 10774819 IC50 = 3500 nM T30082 C4V5XA 10774917 IC50 = 100 nM T30082 C9HZW0 10776513 IC50 > 5000000 nM T30082 CFHV29 10778312 IC50 = 4.58 nM T30082 C2O0RV 10780436 IC50 = 410000 nM T30082 C08YXG 10780715 IC50 = 741.31 nM T30082 CC8R2X 10782665 IC50 = 83000 nM T30082 CK8TJ2 10783430 IC50 = 290 nM T30082 C9PTG2 10785532 IC50 = 47000 nM T30082 C4YS9A 10789991 IC50 = 31030 nM T30082 C2QV9H 10791582 IC50 = 8.6 nM T30082 C90YRE 10792213 IC50 = 8.9 nM T30082 C32WDU 10794714 IC50 = 9772.37 nM T30082 C9YLN1 10799366 IC50 = 134000 nM T30082 CJ8IB2 10801196 IC50 = 5128.61 nM T30082 C2M4JH 10801760 IC50 = 470 nM T30082 C4MFW9 10802453 IC50 = 66 nM T30082 C2IXT8 10807621 Ki = 260 nM T30082 CF0E6N 10811757 IC50 = 40000 nM T30082 CKY87X 10812663 IC50 = 8.9 nM T30082 CKZ53Y 10825928 IC50 = 91000 nM T30082 CDY04M 10830430 IC50 = 13000 nM T30082 CDH9R1 10831927 IC50 = 147 nM T30082 CH7N2T 10836516 IC50 = 5.7 nM T30082 C4FCQ3 10836763 IC50 > 100000 nM T30082 CQ9M1R 10840993 IC50 = 100 nM T30082 CKN2O1 10849613 IC50 = 1000000 nM T30082 C8G6BS 10850978 IC50 = 387.5 nM T30082 CGL0K9 10855014 IC50 = 37.15 nM T30082 CR0C7Z 10858645 IC50 = 20700 nM T30082 CQ9J3V 10859886 IC50 = 16600 nM T30082 C05KRA 10860052 IC50 = 8000 nM T30082 CQY87K 10860441 IC50 = 79.6 nM T30082 C8XSW2 10863593 IC50 = 77624.71 nM T30082 CHF26C 10872974 IC50 = 190 nM T30082 CPF50H 10878304 IC50 = 5.248 nM T30082 CF28NJ 10879668 Ki > 100000 nM T30082 CZH67J 10881476 IC50 = 13900 nM T30082 CKL04Q 10881826 IC50 = 52400 nM T30082 C5IRT2 10893985 IC50 = 30000 nM T30082 C3HZ6S 10894911 IC50 = 120 nM T30082 C1PZ2V 10896395 IC50 = 320 nM T30082 CH49NV 10899196 Ki > 100000 nM T30082 CP93JE 10902085 Ki > 100000 nM T30082 C95XSO 10905408 IC50 = 190 nM T30082 CILE14 10905808 IC50 = 30000 nM T30082 CU4W9S 10909176 IC50 = 77.62 nM T30082 CV35KR 10909236 IC50 = 19.5 nM T30082 CGBH06 10910318 IC50 = 22.91 nM T30082 CSW4G1 10915203 IC50 = 130 nM T30082 CHI85C 10915860 IC50 = 7900 nM T30082 C4M3ZI 10919451 IC50 = 676.08 nM T30082 C3OH9E 10924902 IC50 = 4100 nM T30082 C14OAN 10924975 IC50 = 15400 nM T30082 CR19FE 10927360 IC50 > 10000 nM T30082 C3DSY6 10927599 IC50 = 54.6 nM T30082 CC37RK 10928565 IC50 = 210 nM T30082 CCS2Y7 10941381 IC50 = 56.23 nM T30082 CQ92TC 10941764 IC50 = 3388.44 nM T30082 C0I9NT 10943454 IC50 > 10000 nM T30082 CB7VH2 10945240 IC50 = 54000 nM T30082 C3W0IZ 10950704 IC50 = 50000 nM T30082 CZSC17 10958661 IC50 > 10000 nM T30082 C2Y5XC 10961666 IC50 = 6165.95 nM T30082 C2WRK0 10963725 IC50 = 33.88 nM T30082 CK72HO 10974737 IC50 = 4570.88 nM T30082 C31AFP 10974856 IC50 = 53703.18 nM T30082 CC2F6P 10978630 IC50 = 7800 nM T30082 COJ9N7 10982261 IC50 = 27 nM T30082 CJ7DR2 10985959 IC50 = 11.75 nM T30082 C7BJ5G 10990561 IC50 = 33900 nM T30082 CQ4ZC5 10996738 IC50 = 8.128 nM T30082 C6EZB4 10999994 IC50 = 11000 nM T30082 COVZ49 11001808 IC50 = 30000 nM T30082 C5EO8B 11002266 IC50 = 12200 nM T30082 CN7WQ6 11003427 IC50 = 2000 nM T30082 CI9M6D 11004656 IC50 = 60000 nM T30082 CHLQ20 11004759 IC50 = 2.6 nM T30082 C4NY9F 11006704 IC50 = 27.4 nM T30082 CD96QS 11007082 IC50 = 79.43 nM T30082 C7NZY9 11009341 Ki > 100000 nM T30082 C8V7WK 11010684 IC50 = 280 nM T30082 C60IQT 11011532 IC50 = 79600 nM T30082 CS09JN 11013324 IC50 = 18000 nM T30082 CT5RD0 11014115 IC50 = 30000 nM T30082 C2WD3S 11017037 IC50 = 21.8 nM T30082 C0F1HL 11027759 IC50 = 60000 nM T30082 C4XL5R 11028931 IC50 = 1412.54 nM T30082 C6N9RY 11033566 IC50 = 57900 nM T30082 CX9PC0 11044680 IC50 = 170 nM T30082 CN80QS 11045523 IC50 = 204000 nM T30082 C7JX0P 11047098 IC50 = 82.6 nM T30082 CN6WF9 11051398 IC50 = 17.38 nM T30082 C4MXA8 11055573 IC50 = 850 nM T30082 CM96AO 11058147 IC50 = 320 nM T30082 C46JNI 11068527 IC50 = 3600 nM T30082 CX9GB1 11070319 IC50 = 20000 nM T30082 CQZS78 11071352 IC50 = 6.8 nM T30082 CMY9J6 11076145 IC50 = 35500 nM T30082 CFYX74 11076230 IC50 = 16700 nM T30082 CGOV53 11080189 IC50 = 61 nM T30082 CAQD96 11091137 IC50 = 440 nM T30082 C5ST0C 11097701 IC50 = 160 nM T30082 C7XBI5 11099845 IC50 = 33100 nM T30082 C52YBG 11100067 IC50 = 6000 nM T30082 CPSM68 11104192 IC50 = 204.17 nM T30082 CSYM37 11104646 IC50 = 18.2 nM T30082 CG0UA4 11107589 IC50 = 230 nM T30082 CR8FY3 11108433 IC50 = 1480 nM T30082 C3X4RC 11110155 IC50 = 19100 nM T30082 CF15NS 11113449 IC50 = 6456.54 nM T30082 CJ0RG8 11113852 IC50 = 61659.5 nM T30082 C0J4QW 11113965 IC50 > 100000 nM T30082 CUZ1H3 11114008 IC50 > 30000 nM T30082 C74KUO 11115691 IC50 = 16.6 nM T30082 CEVF09 11119649 IC50 = 6220 nM T30082 CZB4M2 11120913 IC50 = 234000 nM T30082 CJ2P6K 11121264 IC50 > 10000 nM T30082 CST19B 11124861 IC50 = 21.1 nM T30082 CKJ49N 11125225 IC50 = 5754.4 nM T30082 CKRZ24 11125922 IC50 = 10.96 nM T30082 COS32M 11133811 IC50 = 5.4 nM T30082 C1Q5OP 11136870 IC50 = 12.3 nM T30082 C7FPU3 11146640 IC50 = 48.98 nM T30082 CIP41D 11150497 IC50 = 800 nM T30082 C5MKV9 11154961 IC50 = 30199.52 nM T30082 C8FNC1 11156231 IC50 = 147 nM T30082 C9LFS7 11156598 Ki = 0.009 nM T30082 C39DRN 11157463 IC50 = 2.09 nM T30082 CWFE97 11160043 IC50 = 25.12 nM T30082 C7JC9B 11167725 IC50 = 4 nM T30082 CGWM68 11168014 IC50 = 10.9 nM T30082 C8UTA5 11169647 Ki = 1.49 nM T30082 CYL18X 11179973 IC50 = 3.41 nM T30082 C9IV7T 11181553 IC50 = 1071.52 nM T30082 C8YWT1 11188132 IC50 = 8670 nM T30082 C4EU7X 11188905 IC50 = 300 nM T30082 C6L0IS 11190153 IC50 = 1090 nM T30082 CZ2GU4 11191030 IC50 = 95 nM T30082 CBJV46 11192468 IC50 = 2760 nM T30082 CM54US 11192952 IC50 = 4940 nM T30082 CSJ1R4 11193161 IC50 = 60 nM T30082 CH30SU 11204324 IC50 = 1.8 nM T30082 CE21OG 11204682 IC50 = 2630.27 nM T30082 C9EMG6 11209350 IC50 > 50000 nM T30082 CZPB69 11210161 IC50 = 800 nM T30082 CT4Y0D 11210560 IC50 = 1400 nM T30082 CJI9N3 11216927 IC50 = 120.23 nM T30082 C4N9ZL 11221206 IC50 = 500 nM T30082 C93CQK 11221441 IC50 = 2400 nM T30082 C1NI8D 11222968 IC50 > 10000 nM T30082 CY86GP 11226206 IC50 = 6.86 nM T30082 CX6CF4 11232205 IC50 = 50 nM T30082 CEXP98 11233503 IC50 = 2650 nM T30082 CT38EP 11235216 IC50 > 50000 nM T30082 C6TVW3 11238481 IC50 = 10 nM T30082 CSXF65 11238662 IC50 = 75 nM T30082 CV73WE 11239040 IC50 = 79.1 nM T30082 C5FO1B 11243200 IC50 < 10 nM T30082 C6GHQ3 11244670 IC50 > 50000 nM T30082 CC3D2X 11245953 Ki > 100000 nM T30082 CRL20G 11249115 Ki = 0.014 nM T30082 C8GJD2 11249560 IC50 = 0.5 nM T30082 C6LH1M 11250361 IC50 = 44600 nM T30082 CQ1T0O 11253599 IC50 = 4.8 ug.mL-1 T30082 C81GLD 11257074 IC50 = 324 nM T30082 CKTJ19 11260293 IC50 > 30000 nM T30082 CPSO84 11261638 IC50 = 100 nM T30082 C1H0RK 11268352 IC50 = 20417.38 nM T30082 CP6FX1 11268904 IC50 = 100 nM T30082 C2NRQ0 11270327 IC50 > 50000 nM T30082 CEBK83 11272051 IC50 = 46 nM T30082 CC14OZ 11272989 IC50 = 2990 nM T30082 CAP59Z 11278342 IC50 = 56 nM T30082 CSD58O 11280423 Ki > 100000 nM T30082 CYRB74 11283475 Ki = 0.015 nM T30082 C2CQH5 11283831 IC50 = 49600000 nM T30082 CK5SB7 11287987 IC50 = 3000 nM T30082 C1JKX2 11290299 IC50 = 300 nM T30082 CE79LQ 11290672 IC50 = 17 nM T30082 C1KTO4 11301314 IC50 = 2380 nM T30082 CXV91C 11304331 IC50 < 10 nM T30082 CKD79X 11304963 IC50 = 97 nM T30082 CBL8D9 11314048 IC50 > 50000 nM T30082 C91PBQ 11314804 IC50 = 251188.64 nM T30082 CX9JQ2 11316712 IC50 = 6.96 nM T30082 CAJ8O0 11316986 IC50 = 70 nM T30082 C8GX1Y 11322015 Ki > 100000 nM T30082 CO5W9Q 11327297 IC50 > 50000 nM T30082 CEKG13 11329992 IC50 = 1.95 nM T30082 C9JV3E 11330142 Ki = 3.99 nM T30082 C6QVX1 11331507 IC50 = 36.3 nM T30082 CNTY27 11336871 IC50 = 200 nM T30082 C7RJ4Z 11341331 IC50 = 0.5 nM T30082 CG91BA 11350292 IC50 > 50000 nM T30082 CM34HL 11352229 IC50 = 30.1 nM T30082 CAR45P 11359651 IC50 = 26 nM T30082 C59YIW 11359764 IC50 = 302 nM T30082 CK49FX 11364765 IC50 = 80 nM T30082 CSE62M 11365562 IC50 = 520 nM T30082 CZ36FS 11373632 IC50 = 7762.47 nM T30082 CQU73N 11376655 IC50 = 4.1 nM T30082 CI0CV9 11378169 IC50 = 5.754 nM T30082 CIAR80 11380022 IC50 = 360 nM T30082 CPB6X4 11381434 IC50 > 10000 nM T30082 CFS5X7 11382561 IC50 = 330 nM T30082 CSDY73 11385572 IC50 = 35.2 nM T30082 C61VUW 11392125 IC50 = 94 nM T30082 CPNA70 11393196 IC50 = 23 nM T30082 C1YV0R 11393774 IC50 = 83176.38 nM T30082 CJAL17 11397926 IC50 = 18 nM T30082 CWB6K1 11404631 IC50 = 404 nM T30082 C8W9AR 11409935 IC50 = 0.7 nM T30082 CR7E9T 11420352 IC50 = 3700 nM T30082 CXLY31 11425531 IC50 = 830 nM T30082 CL9G3Y 11425872 IC50 = 800 nM T30082 C1JAC5 11425923 Ki = 600 nM T30082 CJPK89 11430659 IC50 = 15848.93 nM T30082 C7T8KU 11432076 Ki = 0.0017 nM T30082 C5DML9 11432727 IC50 = 40 nM T30082 C83YSD 11434003 IC50 = 30902.95 nM T30082 CY72LB 11438752 IC50 = 56 nM T30082 C9BKZ2 11444151 IC50 = 4.4 nM T30082 CL15TO 11445385 IC50 = 3.311 nM T30082 C5TOG0 11445610 Ki = 894 nM T30082 CX8O5K 11446522 IC50 = 199.53 nM T30082 CX1FV3 11449709 IC50 = 12900 nM T30082 CF9M4R 11451482 IC50 = 1100 nM T30082 CS7U9F 11455392 IC50 = 2.9 nM T30082 CY3EG9 11457400 IC50 = 5.754 nM T30082 CKU29D 11461464 IC50 = 13.8 nM T30082 CAE18Q 11464843 IC50 = 1610 nM T30082 C2N7YB 11465667 IC50 = 33 nM T30082 CA92CF 11465956 IC50 = 36 nM T30082 C9E6RY 11478767 Ki = 0.02 nM T30082 C1KBO3 11478903 IC50 = 8 nM T30082 C19ONS 11482774 IC50 = 82 nM T30082 C3WVS4 11489952 Ki = 5.15 nM T30082 CFQ27V 11490183 IC50 = 20 nM T30082 CLD37R 11494779 IC50 > 3000 nM T30082 CSQZ71 11495096 IC50 = 1260 nM T30082 C7OR8M 11504245 IC50 = 0.000005 nM T30082 C6LE2O 11508901 IC50 = 50 nM T30082 C94WCH 11509353 IC50 = 7270 nM T30082 CVN51A 11514475 IC50 = 100 nM T30082 C6ZAT5 11515677 IC50 > 3000 nM T30082 CB6LO5 11515875 IC50 > 3000 nM T30082 C27CVU 11516039 IC50 > 3000 nM T30082 CNQ9H4 11516163 IC50 > 3000 nM T30082 CE34MT 11522221 IC50 > 3000 nM T30082 CA07BP 11530167 IC50 = 142 nM T30082 CSIJ47 11531417 IC50 > 3000 nM T30082 C1YG8Q 11537626 IC50 > 3000 nM T30082 CHLC49 11539744 IC50 = 1410 nM T30082 C3PF8I 11544123 IC50 > 3000 nM T30082 C81ZNF 11545107 IC50 > 3000 nM T30082 C4CA7T 11550697 IC50 = 2420 nM T30082 CF5H2P 11551902 IC50 > 3000 nM T30082 C7I3NU 11555824 IC50 = 0.000005 nM T30082 C80LXZ 11555826 IC50 = 0.000005 nM T30082 C9VAJ6 11555885 IC50 = 0.000005 nM T30082 CH6JG7 11559079 IC50 > 3000 nM T30082 C6B5XD 11561143 IC50 > 3000 nM T30082 C8I2FL 11562215 IC50 = 0.000005 nM T30082 CY9MU1 11563410 IC50 = 0.000005 nM T30082 CYDI05 11565017 IC50 = 58000 nM T30082 C91OHX 11566264 IC50 > 3000 nM T30082 CTX2W5 11566540 IC50 > 3000 nM T30082 C7STM2 11569290 IC50 = 0.000005 nM T30082 C9XNM6 11573923 IC50 = 3430 nM T30082 C3DEL4 11574702 IC50 = 3310 nM T30082 C6P0EV 11576166 IC50 = 17000 nM T30082 CH04PB 11588880 IC50 = 3550 nM T30082 C5AN1O 11589433 IC50 > 3000 nM T30082 CXO0Z9 11590581 IC50 = 0.000005 nM T30082 C5DUX1 11593477 IC50 = 69.18 nM T30082 C96RTF 11595013 IC50 = 97 nM T30082 C19WSH 11595694 IC50 > 3000 nM T30082 C2C4KA 11599119 IC50 = 0.1 nM T30082 CK2PB1 11603489 IC50 = 1420 nM T30082 CIJ6B4 11603744 IC50 > 3000 nM T30082 CLOD63 11606144 IC50 = 0.87 nM T30082 CH6ZB0 11610321 IC50 > 3000 nM T30082 CCS65Q 11610402 IC50 = 190 nM T30082 COAU76 11620371 IC50 = 0.000005 nM T30082 CAF5O0 11625278 IC50 = 273 nM T30082 C2LD0Q 11631221 IC50 = 38 nM T30082 CV5RH1 11631680 IC50 = 5510 nM T30082 CEY1C7 11645534 IC50 = 20 nM T30082 C95XBL 11645797 IC50 > 3000 nM T30082 CFB27N 11646207 IC50 > 3000 nM T30082 CQX1I8 11647230 IC50 = 25200 nM T30082 CBGT09 11648619 IC50 = 0.23 nM T30082 CZ0I7M 11652422 IC50 > 3000 nM T30082 C8E1TB 11652860 IC50 > 3000 nM T30082 CZ1LE6 11659857 IC50 > 3000 nM T30082 CT61SY 11661034 IC50 > 3000 nM T30082 CCZU50 11661185 IC50 > 3000 nM T30082 CU1K8W 11666118 IC50 = 486 nM T30082 CO3EB9 11666940 IC50 > 3000 nM T30082 C8E6NF 11669798 IC50 = 180 nM T30082 C0AR9Z 11681391 IC50 = 36 nM T30082 CI5MT9 11681880 IC50 = 6700 nM T30082 C1PRY4 11682031 IC50 > 3000 nM T30082 CE1Z3R 11682380 IC50 > 3000 nM T30082 C5QXE9 11688419 IC50 > 3000 nM T30082 CWBC32 11689439 IC50 > 3000 nM T30082 CC1ZN6 11694595 IC50 = 610 nM T30082 CR1IW0 11697764 IC50 = 30 nM T30082 C5HYV7 11698149 IC50 = 256 nM T30082 CJ6UR7 11706508 IC50 = 0.000005 nM T30082 CB39ON 11709265 IC50 = 7 nM T30082 C71EWN 11713155 IC50 = 0.000005 nM T30082 CJPM86 11722402 IC50 > 20000 nM T30082 C5FJ0D 11722860 IC50 = 22.1 nM T30082 CNI0S1 11726118 IC50 = 10000 nM T30082 CL2O3H 11726428 IC50 = 43 nM T30082 C5UQT1 11728283 IC50 > 100000 nM T30082 C63THL 11731635 IC50 = 6300 nM T30082 CZ2S3H 11734156 IC50 = 11.7 nM T30082 C45PDY 11734220 IC50 = 46000 nM T30082 CBY03I 11739675 IC50 = 4300 nM T30082 C2I0ZL 11740281 IC50 = 24 nM T30082 CA8G0C 11740282 IC50 = 125 nM T30082 C3W5JF 11740877 IC50 = 21 nM T30082 CK57XI 11741146 IC50 = 127 nM T30082 CM9W1N 11741355 IC50 = 145 nM T30082 CVMA06 11742091 IC50 = 55200 nM T30082 CWD05H 11743869 IC50 = 10.1 nM T30082 C1SDF0 11752376 IC50 = 32.7 nM T30082 C51RYW 11752643 IC50 = 3 nM T30082 CLMV71 11753218 Ki = 13.37 nM T30082 CAMR83 11753295 IC50 = 21.9 nM T30082 CF70QL 11755538 IC50 > 100000 nM T30082 CTN3A2 11756147 IC50 = 3500 nM T30082 CB8A6W 11762106 IC50 = 14 nM T30082 CQB14T 11763573 IC50 = 9810 nM T30082 C7MFV8 11763757 IC50 = 134.9 nM T30082 C7OPQ0 11772375 IC50 = 200 nM T30082 CIRW35 11773139 IC50 = 48977.88 nM T30082 CV84AY 11776726 IC50 = 10.9 nM T30082 CIQ7A4 11777992 IC50 = 1000 nM T30082 CV4W8C 11784091 IC50 = 470 nM T30082 CZRE80 11786613 IC50 = 137000 nM T30082 CG34JX 11792247 IC50 = 780.4 nM T30082 CQ6YH2 11799236 IC50 = 41130 nM T30082 CS23AV 11800047 IC50 = 37.4 nM T30082 C7Q8DE 11800701 IC50 = 2.8 nM T30082 CCQN45 11805526 Ki > 100000 nM T30082 CCUJ91 11808166 IC50 = 220 nM T30082 C7WYG3 11810853 IC50 = 710 nM T30082 C7MEZ0 11811901 IC50 = 25000 nM T30082 CX97ZV 11814517 IC50 = 112.2 nM T30082 CUYD78 11821709 IC50 = 3240 nM T30082 C0GC9X 11822595 IC50 = 540 nM T30082 C85DZW 11824488 IC50 = 11000 nM T30082 C47XTS 11825091 IC50 = 3400 nM T30082 C2OJ4S 11825837 IC50 = 430 nM T30082 CNA09T 11826485 IC50 = 80000 nM T30082 C6TMU5 11833388 IC50 = 30200 nM T30082 C0CR2G 11848185 IC50 > 200000 nM T30082 CVS5N8 11854653 IC50 = 386 nM T30082 CS85HX 11948486 IC50 > 1000000 nM T30082 C2S9XC 11957509 IC50 = 3370 nM T30082 CODF94 12050842 IC50 = 130000 nM T30082 CTM34I 12109666 IC50 = 91070 nM T30082 CJC3N0 12146686 IC50 = 3700 nM T30082 C6F3ZN 12176878 IC50 = 172.1 nM T30082 C7RZY1 12176883 IC50 = 56.9 nM T30082 CKG7A0 12222796 Ki > 100000 nM T30082 CC3MQ9 12314224 IC50 = 56 nM T30082 C1RID4 12327577 IC50 > 20000 nM T30082 C6SB2O 12344042 IC50 = 500 nM T30082 CWQD79 12624603 IC50 = 456000 nM T30082 C4J3SD 12624606 IC50 = 270600 nM T30082 CE1G4B 12927714 IC50 = 3000 nM T30082 CC3U2F 12927716 IC50 > 10000 nM T30082 C5L0GN 12927905 IC50 = 2290000 nM T30082 C48RAC 12989874 IC50 = 590 nM T30082 C1R4MF 12995052 IC50 = 560 nM T30082 C54QHI 13006034 IC50 = 140 nM T30082 C6XHS1 13006035 IC50 = 14 nM T30082 CG7AZ9 13006036 IC50 = 28 nM T30082 CDP08C 13006037 IC50 = 23 nM T30082 C0AH2N 13006038 IC50 = 31 nM T30082 CIY8G4 13006039 IC50 = 78 nM T30082 CTX5Q6 13006040 IC50 = 26 nM T30082 CJ43VT 13006041 IC50 = 285 nM T30082 CS7V4K 13006042 IC50 = 260 nM T30082 CT5C2K 13006043 IC50 = 1300 nM T30082 CH46IX 13006044 IC50 = 1500 nM T30082 C3VSW6 13006045 IC50 = 15 nM T30082 CFE3W8 13006046 IC50 = 780.4 nM T30082 CU0BN1 13006047 IC50 > 10000 nM T30082 CAJG53 13300537 IC50 = 12000 nM T30082 C0KSR2 13497076 IC50 = 720000 nM T30082 CEO81S 13552185 IC50 = 654000 nM T30082 CL4MK3 13552226 IC50 = 1270000 nM T30082 CC4AI3 13582542 IC50 = 12890 nM T30082 C7PST2 13692942 IC50 = 12.02 nM T30082 C4TA0V 13735450 IC50 = 1700 nM T30082 C8B5LO 13780062 Ki > 100000 nM T30082 C3YOX2 13827082 Ki > 100000 nM T30082 C4CR1L 13827083 Ki > 100000 nM T30082 CK08BO 13896866 IC50 > 500000 nM T30082 C0TRN9 13934286 IC50 = 26780 nM T30082 CO5V8C 13969569 IC50 = 970 nM T30082 CYJI38 13970960 IC50 = 81500 nM T30082 C7MV6G 13997263 IC50 > 100000 nM T30082 CU2M9R 14107712 IC50 = 9887 nM T30082 C4YBN3 14109375 IC50 = 24040 nM T30082 C2G8DC 14157083 IC50 = 597035.29 nM T30082 C6P1EB 14157085 IC50 = 470977.33 nM T30082 CJS4R6 14193572 IC50 = 330 nM T30082 CM6R4N 14193573 IC50 = 21 nM T30082 C39VGI 14193575 IC50 = 32 nM T30082 C6BP1S 14193577 IC50 = 150 nM T30082 C5HUP2 14318563 IC50 = 9200 nM T30082 CDBY65 14318564 IC50 = 13510 nM T30082 C0PO5M 14349781 IC50 = 785 nM T30082 C7NE3Y 14372818 IC50 = 31.5 nM T30082 CXY61Q 14372820 IC50 = 1096.48 nM T30082 CGJ4B5 14372825 IC50 = 10000 nM T30082 C8HST3 14372826 IC50 = 455 nM T30082 C8XY5F 14372827 IC50 = 1120 nM T30082 C6O3QW 14372830 IC50 = 2600 nM T30082 CSU1C6 14372831 IC50 = 429 nM T30082 CVI4B2 14372832 IC50 = 6309.57 nM T30082 CDW0M2 14372833 IC50 = 42 nM T30082 CJN71L 14491727 IC50 = 263.03 nM T30082 CTB5H2 14539882 Ki = 3100 nM T30082 CV7A3W 14539951 IC50 = 109200 nM T30082 CULX32 14553493 IC50 = 411 nM T30082 CSGJ12 14553576 IC50 = 1540 nM T30082 CWO74N 14553581 IC50 = 755 nM T30082 CH27JR 14609844 IC50 = 3312 nM T30082 C93MXE 14735915 IC50 = 14000 nM T30082 CAH47C 14735925 IC50 = 20000 nM T30082 C3VX2W 14783860 IC50 = 560 nM T30082 CMB2L4 14847270 IC50 = 96800 nM T30082 C3KTU6 14857744 IC50 = 169 nM T30082 C1XBP2 14857745 IC50 = 159 nM T30082 CPY1W8 14857746 IC50 = 206 nM T30082 CP4Q3I 14857748 IC50 = 171 nM T30082 CPS8V3 14857750 IC50 = 72 nM T30082 CLG16Z 14857751 IC50 = 143 nM T30082 CMF7U1 14877070 IC50 = 70000 nM T30082 CP25BA 14985958 IC50 = 3300 nM T30082 CQWN41 14997887 IC50 = 1.318 nM T30082 CW1YL6 14997888 IC50 = 6.31 nM T30082 CKCA80 14997889 IC50 = 7.079 nM T30082 C6EA9P 14997890 IC50 = 8.913 nM T30082 C98IZW 14997891 IC50 = 13.18 nM T30082 CG91HZ 14997892 IC50 = 19.95 nM T30082 C7QT0X 14997893 IC50 = 380 nM T30082 C6XL3Y 14997894 IC50 = 380 nM T30082 C0X4PT 15005007 IC50 = 2100 nM T30082 CH9PO3 15005008 IC50 = 1200 nM T30082 CK69GO 15005009 IC50 = 650 nM T30082 C6V9HJ 15005010 IC50 = 270 nM T30082 C1EQ0S 15043261 IC50 = 229086.77 nM T30082 C8PYV9 15043264 IC50 = 181970.09 nM T30082 CL2C7Y 15044210 Ki > 100000 nM T30082 CNJ2A9 15085436 IC50 = 350 nM T30082 C73XRZ 15108314 IC50 = 240000 nM T30082 CJ3E7T 15125273 IC50 = 260 nM T30082 CA13LZ 15125274 IC50 = 337 nM T30082 C9WTF1 15125278 IC50 = 362 nM T30082 C3ZXK7 15150646 IC50 = 263 nM T30082 CU4Z1T 15153347 IC50 = 5.3 nM T30082 C8JI6S 15153348 IC50 = 7.7 nM T30082 CJX1E3 15153349 IC50 = 8.4 nM T30082 CF3Y2O 15153350 IC50 = 94 nM T30082 CEA9O6 15153351 IC50 = 480 nM T30082 CR81ZV 15153352 IC50 = 4400 nM T30082 CI81BH 15153353 IC50 = 1200 nM T30082 C9N8AZ 15153354 IC50 = 0.9 nM T30082 CL1QB6 15153356 IC50 = 1.5 nM T30082 CQV1E5 15153357 IC50 = 0.82 nM T30082 C5KXT4 15153359 IC50 = 8.9 nM T30082 CFNI61 15153360 IC50 = 160 nM T30082 CXC83S 15153361 IC50 = 2900 nM T30082 CR1N2D 15153362 IC50 = 180 nM T30082 CZ4TU3 15164572 IC50 = 3000 nM T30082 C8NDO3 15164573 IC50 = 48000 nM T30082 CWZC62 15164575 IC50 = 2500 nM T30082 C7JMR1 15164576 IC50 = 44000 nM T30082 CX2C0Y 15164578 IC50 = 9000 nM T30082 CH96CL 15164579 IC50 = 1500 nM T30082 CR8XS3 15164580 IC50 = 1300 nM T30082 C2AV5N 15249928 IC50 = 1000 nM T30082 C2R3EJ 15270569 IC50 = 114.4 nM T30082 C65LFC 15337793 IC50 = 1700 nM T30082 CDW8F0 15337794 IC50 = 1500 nM T30082 CEJ8R4 15337804 IC50 < 100000 nM T30082 C3L5XF 15337805 IC50 = 1260 nM T30082 CM6O0G 15340688 IC50 = 3.4 nM T30082 C7ITH5 15340689 EC50 = 12 nM T30082 CZ3WJ2 15490813 IC50 = 115 nM T30082 C20BEI 15552341 IC50 = 39.81 nM T30082 CF83ID 15625290 IC50 = 2500 nM T30082 C1S6GM 15720175 IC50 = 3860 nM T30082 CB02SK 15745369 IC50 = 268.8 nM T30082 CHG23X 15751376 IC50 = 58 nM T30082 CM9CZ4 15751381 IC50 = 20 nM T30082 C4MH9V 15751383 IC50 = 233 nM T30082 CR2M7V 15751409 IC50 = 1076 nM T30082 C60XWP 15751411 IC50 = 2192 nM T30082 CL0NC5 15751413 IC50 = 253 nM T30082 CHD8B2 15751415 IC50 = 629 nM T30082 C9X6VS 15751417 IC50 = 546 nM T30082 CVH65O 15984120 IC50 = 21 nM T30082 C9GNW0 16086577 IC50 > 10 ug.mL-1 T30082 CR2J0F 16094841 IC50 = 365 nM T30082 C34FJR 16094854 IC50 = 89.2 nM T30082 C8JM2I 16094855 IC50 = 241 nM T30082 CCL15D 16094856 IC50 = 18.2 nM T30082 COID78 16094857 IC50 = 5.24 nM T30082 CMT73Z 16094858 IC50 = 135 nM T30082 C3RN7X 16094859 IC50 = 72.1 nM T30082 CWI3K1 16094860 IC50 = 8.39 nM T30082 CG14KR 16094871 IC50 = 51.6 nM T30082 CKJ3F6 16094872 IC50 = 17 nM T30082 CD9S2E 16094873 IC50 = 5.65 nM T30082 C35HXC 16094875 IC50 = 40.7 nM T30082 CU8W5V 16094876 IC50 = 59 nM T30082 CB3O6A 16212317 IC50 = 1690 nM T30082 C28IBN 16219608 IC50 = 210 nM T30082 C6GD9H 16235993 IC50 = 1800 nM T30082 CG5J7B 16584800 IC50 < 600000 nM T30082 C7MSU0 16653132 IC50 > 100000 nM T30082 C9S4KN 16666409 IC50 = 8500 nM T30082 CX0H5Q 16680726 IC50 = 3800 nM T30082 CBE91C 16726036 IC50 = 68800 nM T30082 CH9Y5B 17159064 IC50 = 620 nM T30082 C5ZMI9 17159212 IC50 = 2200 nM T30082 CF6ZW1 17159244 IC50 = 2200 nM T30082 C80YMT 17159252 IC50 = 720 nM T30082 CO02WZ 17387125 IC50 = 110000 nM T30082 CZ26EM 17680296 IC50 = 204.17 nM T30082 C2OF8S 18471933 Ki > 100000 nM T30082 CD6NW8 18992275 IC50 = 158.49 nM T30082 C67KIN 19108449 IC50 = 25.12 nM T30082 C39VUS 19760985 IC50 = 14240 nM T30082 CYP5J8 19770286 IC50 = 78 nM T30082 C7Y4FO 19770289 IC50 = 99 nM T30082 CO7R0C 19770292 IC50 = 615 nM T30082 CW0H1Y 20055993 IC50 = 22970 nM T30082 CY20PU 20081899 IC50 = 4.467 nM T30082 C2ZNO6 20186976 Ki = 160 nM T30082 C45TLN 21204337 IC50 = 1310000 nM T30082 C0ET8M 21362734 IC50 > 10000 nM T30082 C72BMS 21409569 IC50 = 5400 nM T30082 CB1U4Z 21589046 IC50 = 56.7 nM T30082 CQKH16 21592283 IC50 = 25910 nM T30082 CK0YE8 21607150 IC50 = 48500 nM T30082 CJKR07 21632954 IC50 = 30260 nM T30082 CEJ49C 21633084 IC50 = 17140 nM T30082 C2FBA3 21672659 IC50 > 30000 nM T30082 CX8W6N 21839636 IC50 = 37.8 nM T30082 CT3YN1 21839638 IC50 = 35.4 nM T30082 C5GZ1L 21839640 IC50 = 2.11 nM T30082 C8YO3H 21839642 IC50 = 29.5 nM T30082 CWR90B 21839649 IC50 = 51.6 nM T30082 CI29XS 22064898 IC50 > 100000 nM T30082 C1NOW2 22197665 IC50 = 10 nM T30082 CM3Y1I 22574246 Ki > 100000 nM T30082 C0F6KD 22782067 IC50 = 71000 nM T30082 C5IZQ8 23093594 IC50 = 400 nM T30082 C7KCD5 23247894 IC50 = 18350 nM T30082 CK15SO 23448959 IC50 = 147 nM T30082 C13RZX 23624871 IC50 = 42.5 nM T30082 C6SY8I 23634493 Ki = 453.15 nM T30082 CSK7Z4 23634753 IC50 = 351 nM T30082 C1S9XV 23634999 IC50 = 839 nM T30082 C15ASX 23635398 IC50 > 50000 nM T30082 C9F1MQ 23635399 IC50 > 50000 nM T30082 CXIA45 23635400 IC50 > 50000 nM T30082 CQ0H4M 23635401 IC50 > 50000 nM T30082 CMT2D6 23635496 IC50 = 517 nM T30082 CZ5R6B 23635511 IC50 > 50000 nM T30082 C5S2QB 23635512 IC50 > 50000 nM T30082 C4B8MX 23635513 IC50 > 50000 nM T30082 CWD7J8 23635514 IC50 > 50000 nM T30082 C0ASM1 23635515 IC50 > 50000 nM T30082 CKP70J 23635516 IC50 > 50000 nM T30082 CM0X3T 23635632 IC50 > 50000 nM T30082 C0VL9W 23635633 IC50 > 50000 nM T30082 CJ73KM 23635634 IC50 > 50000 nM T30082 CWI26H 23635635 IC50 > 50000 nM T30082 C4GA2J 23635637 IC50 > 50000 nM T30082 C1P7GL 23635748 IC50 = 5242 nM T30082 CV8QU5 23635749 IC50 = 265 nM T30082 CT46CR 23635766 IC50 > 50000 nM T30082 CVJ6C0 23635767 IC50 > 50000 nM T30082 CU61DC 23635768 IC50 > 50000 nM T30082 CF91IH 23635891 IC50 > 50000 nM T30082 CT67MK 23635892 IC50 > 50000 nM T30082 CKM0C8 23635893 IC50 > 50000 nM T30082 CC1PX4 23635894 IC50 > 50000 nM T30082 C0XQ8E 23635895 IC50 > 50000 nM T30082 CCPS26 23635896 IC50 > 50000 nM T30082 C4UY7R 23636019 IC50 > 50000 nM T30082 CHTN58 23636020 IC50 > 50000 nM T30082 CPV52Y 23636021 IC50 > 50000 nM T30082 CD71KA 23636022 IC50 > 50000 nM T30082 CXP7U0 23642826 IC50 = 113000 nM T30082 C4NE7D 23642915 IC50 = 2320 nM T30082 C93CLQ 23644605 IC50 = 1.6 nM T30082 CB9V7K 23644606 IC50 = 28840.32 nM T30082 CMH24N 23644647 IC50 = 0.82 nM T30082 CQ49JO 23644649 IC50 = 0.33 nM T30082 C4HV8T 23644653 IC50 = 0.4 nM T30082 C01OPD 23644658 IC50 = 27 nM T30082 CWL64B 23644773 IC50 = 1584.89 nM T30082 CSQ9L7 23644774 IC50 = 75 nM T30082 C3AS4O 23644775 IC50 = 22 nM T30082 C2V8TA 23644776 IC50 = 0.9 nM T30082 C5W0NY 23644777 IC50 = 0.6 nM T30082 C8YQA2 23644778 IC50 = 4.8 nM T30082 CPO4L8 23644779 IC50 = 1.3 nM T30082 CSU1T2 23644780 IC50 = 1.9 nM T30082 CZH24F 23644782 IC50 = 2.7 nM T30082 C56IML 23644785 IC50 = 1202.26 nM T30082 C2UK1G 23644786 IC50 = 1659.59 nM T30082 C5OJP1 23644790 IC50 = 5888.44 nM T30082 CQ6DC0 23644791 IC50 = 67608.3 nM T30082 CAJ0V1 23644792 IC50 = 6606.93 nM T30082 CQH18E 23644793 IC50 = 6456.54 nM T30082 CO58YI 23644794 IC50 = 4265.8 nM T30082 CY4J7F 23644795 IC50 = 3890.45 nM T30082 CJM39K 23644796 IC50 = 4570.88 nM T30082 CG07CB 23644797 IC50 = 5370.32 nM T30082 CM39BI 23645223 IC50 = 38.4 nM T30082 CW8F0V 23645224 IC50 = 21.5 nM T30082 CTW9J8 23645267 IC50 = 0.5 nM T30082 CRB3O6 23645269 IC50 = 0.34 nM T30082 CB8H9A 23645271 IC50 = 0.45 nM T30082 C34ZIH 23645273 IC50 = 0.33 nM T30082 CK2NJ4 23645289 IC50 = 13 nM T30082 CA3P8O 23645310 IC50 = 30 nM T30082 C5B2OL 23645311 IC50 = 6140 nM T30082 C2QFC7 23645314 IC50 = 31800 nM T30082 CRC6A7 23645315 IC50 = 34900 nM T30082 CY3LE0 23645319 IC50 = 525000 nM T30082 C3XDF8 23657682 IC50 = 7.61 nM T30082 CHKQ18 23657684 IC50 = 15.8 nM T30082 C6WY3U 23669322 Ki > 100000 nM T30082 CG61EZ 23765385 IC50 = 7500 nM T30082 C4R5ET 24192080 IC50 = 37000 nM T30082 C8TQC7 24276654 IC50 = 42000 nM T30082 C5CS6H 24276655 IC50 = 379000 nM T30082 C75MBH 24276662 IC50 = 61400 nM T30082 CA1CP6 24276664 IC50 = 275300 nM T30082 C4GRE7 24276682 IC50 = 321000 nM T30082 CDGZ60 24276683 IC50 = 381000 nM T30082 CBXC05 24424330 IC50 = 520 nM T30082 CANS31 24749809 IC50 = 1.83 nM T30082 C4Z2EB 24749810 IC50 = 19.7 nM T30082 C4FVB7 24749811 IC50 = 6.65 nM T30082 CZRW61 24796898 IC50 = 18060 nM T30082 CO9D4U 24799948 IC50 = 69.5 nM T30082 C6LV5R 24799949 IC50 = 21.6 nM T30082 C8JPO2 24800125 IC50 = 93 nM T30082 C64FMN 24800126 IC50 = 10 nM T30082 C8GKX5 24800127 IC50 = 6.3 nM T30082 C6DSC8 24800128 IC50 = 5.6 nM T30082 CW7LB1 24800129 IC50 = 35.5 nM T30082 CZ14LB 24800130 IC50 = 28.2 nM T30082 C59BPF 24800294 IC50 = 22.6 nM T30082 C07CZO 24800295 IC50 = 45.7 nM T30082 C5H3EC 24800296 IC50 = 6.4 nM T30082 C0QLV7 24800297 IC50 = 11.1 nM T30082 CAO8P0 24800298 IC50 = 18.1 nM T30082 CARE83 24800299 IC50 = 50.7 nM T30082 CZ0GN5 24800469 IC50 = 226 nM T30082 CQNB75 24825630 Ki > 100000 nM T30082 C2NQ6G 24825767 IC50 = 316.23 nM T30082 CF6W3Z 24833568 IC50 = 0.7 nM T30082 CVZ3G8 24845717 IC50 = 15 nM T30082 CMF3P2 24845873 IC50 = 4000 nM T30082 CT78NC 24854122 IC50 = 92400 nM T30082 CWHK93 24854124 IC50 = 31900 nM T30082 CR6M2L 24863097 Ki = 0.0118 nM T30082 CBP1Y5 24865177 IC50 = 32600 nM T30082 COR9K5 24865178 IC50 = 17400 nM T30082 CIY6F4 24865179 IC50 = 40700 nM T30082 CKB7T5 24865359 IC50 = 127000 nM T30082 CS1VB7 24865360 IC50 = 10500 nM T30082 C50JUL 24865361 IC50 = 127000 nM T30082 CH0WZ8 24865362 IC50 = 281000 nM T30082 C9W8TE 24865363 IC50 = 177000 nM T30082 C2CX0D 24879253 Ki = 2.672 nM T30082 CO3D6F 24879256 Ki = 0.1191 nM T30082 CE7RA8 24879313 Ki = 1.718 nM T30082 COVB34 24879315 Ki = 1.63 nM T30082 CX60OH 24879317 Ki = 20.88 nM T30082 CW49DK 24879319 Ki = 0.223 nM T30082 C3DGL7 24879377 Ki = 0.162 nM T30082 CQM5Y4 24879379 Ki = 0.0847 nM T30082 CA6WB0 24879381 Ki = 0.1359 nM T30082 CRWB78 24879383 Ki = 0.768 nM T30082 C3GTP2 24879451 Ki = 7.45 nM T30082 CDI31X 24879453 Ki = 13.27 nM T30082 C51PQF 24881876 IC50 = 0.88 nM T30082 CLM2P5 24881945 IC50 = 5.13 nM T30082 CDI95B 24881949 IC50 = 2.16 nM T30082 CLW51O 24936061 IC50 = 7.16 nM T30082 CABV24 24936088 Ki = 64400 nM T30082 CO1ID8 24949376 IC50 = 2.15 nM T30082 C5VL9C 24949523 IC50 = 1.65 nM T30082 C2UZ4A 24949524 IC50 = 1.54 nM T30082 C3OV2G 24949525 IC50 = 2.57 nM T30082 CIT46H 24994026 IC50 = 0.27 nM T30082 CDY49T 25016412 IC50 = 24200 nM T30082 CVQY09 25016666 IC50 = 48500 nM T30082 CAVC47 25033601 IC50 = 8100 nM T30082 CB5U1A 25135608 IC50 = 880000 nM T30082 C7JY8N 25135721 IC50 = 2477.42 nM T30082 CI9HU8 25135723 IC50 = 2950000 nM T30082 C0BT7H 25135724 IC50 = 2792.54 nM T30082 CHIR40 25135837 IC50 = 510000 nM T30082 CLMS71 25135964 IC50 = 5584.7 nM T30082 CLIB48 25136381 IC50 = 5727.96 nM T30082 CYT6K0 25137488 IC50 = 35000 nM T30082 C4W1QB 25137489 IC50 = 3000 nM T30082 CHJ67F 25137491 IC50 = 70000 nM T30082 CV73ZD 25137492 IC50 = 30000 nM T30082 C2RX3Y 25137493 IC50 = 6000 nM T30082 CUC8N5 25141405 IC50 > 100000 nM T30082 CHN93D 25145301 IC50 = 7800 nM T30082 C3P4KA 25149263 IC50 = 15.9 nM T30082 CX50VY 25149264 IC50 = 14 nM T30082 CU45TK 25149265 IC50 = 0.37 nM T30082 CU7EV3 25149453 IC50 = 25.7 nM T30082 CB9Q1Y 25149538 IC50 = 4.83 nM T30082 CEF4M1 25150256 IC50 = 4160 nM T30082 CES10Z 25150257 IC50 = 8550 nM T30082 CW5Y9S 25150356 IC50 = 68.9 nM T30082 C6KSF0 25150451 IC50 = 1.41 nM T30082 CEL09B 25150452 IC50 = 72.4 nM T30082 CKW2Z0 25150453 IC50 = 7.7 nM T30082 CB7K2G 25150454 IC50 = 53.5 nM T30082 CZ47PT 25168164 IC50 = 1000 nM T30082 CMYQ85 25168165 IC50 = 2511.89 nM T30082 C42VOK 25168166 IC50 = 1258.93 nM T30082 CB5A1G 25197363 Ki = 62.25 nM T30082 CRN1B6 25197364 Ki = 616.7 nM T30082 C3BY8I 25197494 Ki = 235.5 nM T30082 CY7MW6 25197495 Ki = 919.62 nM T30082 C15JXP 25197497 Ki = 236.52 nM T30082 C0Q6PW 25197628 Ki = 126.75 nM T30082 CJ7H5C 25197629 Ki = 198.49 nM T30082 CPCX38 25197632 Ki = 70.9 nM T30082 CSX7D4 25197633 Ki = 95.21 nM T30082 CRS17Z 25197760 Ki = 524.99 nM T30082 C57ATH 25197761 Ki = 161.03 nM T30082 CRM14V 25197762 Ki = 506.78 nM T30082 CBN1H2 25197763 Ki = 918.25 nM T30082 CMZ46C 25197765 Ki = 21.66 nM T30082 CM9PV8 25197906 Ki = 22.28 nM T30082 C8A9UF 25197907 Ki = 772.65 nM T30082 C4GV3H 25197910 Ki = 59.34 nM T30082 CVL46O 25198054 Ki = 1040 nM T30082 C3R1LE 25198055 Ki = 73.78 nM T30082 CSLH31 25204947 IC50 = 131 nM T30082 C9NG2M 25205011 IC50 = 508 nM T30082 C0TWB6 25211256 Ki = 0.08 nM T30082 CRKA79 25221268 IC50 > 20000 nM T30082 C8IQC1 27764355 IC50 = 368 nM T30082 CL89DY 35793912 IC50 = 680 nM T30082 CKJ82C 38864639 IC50 > 100000 nM T30082 CH4UY3 41474021 IC50 > 100000 nM T30082 CJ06DE 42597801 IC50 = 460 nM T30082 C39RQM 42597802 IC50 = 345000 nM T30082 CL70RY 42597803 IC50 = 36800 nM T30082 CJX2O8 42598036 IC50 = 2370 nM T30082 C59KBA 42598037 IC50 = 27200 nM T30082 CEK7A5 42598038 IC50 = 54000 nM T30082 CX4H1M 42598039 IC50 = 4270 nM T30082 C7GO1F 42598040 IC50 = 3710 nM T30082 CE6Y3Z 42598041 IC50 = 1650 nM T30082 C0X7NH 42598042 IC50 = 570 nM T30082 CNGR23 42598273 IC50 = 1410 nM T30082 C8K3WA 42598274 IC50 = 2100 nM T30082 CF75TP 42598275 IC50 = 1570 nM T30082 CXZ19Y 42598510 IC50 = 8640 nM T30082 CBOI16 42598737 IC50 = 1820 nM T30082 CT0N9J 42598738 IC50 = 19600 nM T30082 C2UN9H 42618134 IC50 = 226 nM T30082 CH6X2V 42618135 IC50 = 71 nM T30082 CCAU57 42618136 IC50 = 45 nM T30082 C0EO3S 42618137 IC50 = 158 nM T30082 CH21YS 42618138 IC50 = 223 nM T30082 C2D4GJ 42637909 IC50 = 36 nM T30082 CE4Q1Z 42637910 IC50 = 378 nM T30082 CXM1J2 43802807 IC50 = 358200 nM T30082 CA6I9J 43802854 IC50 = 394000 nM T30082 C5AYT4 43802949 IC50 = 478000 nM T30082 C10NIO 43803032 IC50 = 363000 nM T30082 C1E5GI 43824597 IC50 = 4100 nM T30082 CEPY38 43826154 IC50 = 199.5 nM T30082 C2ZDR5 44123701 IC50 = 93 nM T30082 CN6GY5 44178775 IC50 = 20 nM T30082 C7YR8O 44224102 IC50 = 19.3 nM T30082 CMQ73T 44241603 IC50 = 6.75 nM T30082 CPS81V 44245423 IC50 = 185 nM T30082 C4Q2KU 44245424 IC50 = 90 nM T30082 CNME62 44247959 IC50 = 9.64 nM T30082 CUP1V5 44275223 IC50 = 13000 nM T30082 CZE8D6 44281107 IC50 = 12487 nM T30082 CE9WL8 44281141 IC50 = 506 nM T30082 CR9OD5 44281155 IC50 = 93 nM T30082 CN8PV5 44281161 IC50 = 176 nM T30082 C37CIM 44281162 IC50 = 20 nM T30082 COY3Z8 44281181 IC50 = 546 nM T30082 CPJ4S3 44281212 IC50 = 1076 nM T30082 C5DVP0 44281226 IC50 = 208 nM T30082 CFG32T 44281227 IC50 = 69 nM T30082 C2P0WU 44281240 IC50 = 1330 nM T30082 CCV58N 44281253 IC50 = 629 nM T30082 COP30Z 44281256 IC50 = 253 nM T30082 C5S8AK 44281257 IC50 = 2192 nM T30082 CP0W7V 44281393 IC50 = 154 nM T30082 CUM98A 44281438 IC50 = 90 nM T30082 CMD43R 44281439 IC50 = 381 nM T30082 C7CVS3 44281456 IC50 = 38 nM T30082 CN8U6W 44281478 IC50 = 77 nM T30082 CQR91O 44281479 IC50 = 114 nM T30082 CWI3J4 44298002 IC50 = 550 nM T30082 C3O4PU 44300866 IC50 = 2000 nM T30082 C0EY7K 44300875 IC50 = 3000 nM T30082 CD41KT 44301330 IC50 > 10000 nM T30082 CJA2T0 44301335 IC50 > 10000 nM T30082 CX6R5B 44301337 IC50 > 10000 nM T30082 CAC96R 44301339 IC50 > 10000 nM T30082 C5XJR3 44301392 IC50 > 10000 nM T30082 CLH16N 44301394 IC50 > 10000 nM T30082 CC02KE 44301404 IC50 > 10000 nM T30082 CK65ZA 44301406 IC50 > 10000 nM T30082 CBOU57 44301457 IC50 > 10000 nM T30082 CVK47A 44301459 IC50 > 10000 nM T30082 CIV9U5 44301473 IC50 > 10000 nM T30082 C3G9WE 44301475 IC50 > 10000 nM T30082 C3J1VA 44301478 IC50 > 10000 nM T30082 C7CUT9 44301484 IC50 > 10000 nM T30082 CQVZ61 44301486 IC50 = 10000 nM T30082 CM7U0C 44301488 IC50 = 330 nM T30082 C2TZF5 44301490 IC50 = 10000 nM T30082 C7I6FJ 44301496 IC50 > 10000 nM T30082 CUR93P 44301498 IC50 = 10000 nM T30082 CW5UF3 44301500 IC50 > 10000 nM T30082 C2J8HA 44301574 IC50 > 10000 nM T30082 CVHZ92 44301613 IC50 > 10000 nM T30082 C1DIX5 44301615 IC50 > 10000 nM T30082 CZSQ09 44301633 IC50 > 10000 nM T30082 CXO36Q 44301667 IC50 = 1040 nM T30082 C2KEH6 44301669 IC50 > 10000 nM T30082 C6QJC1 44301671 IC50 = 10000 nM T30082 C1PMV7 44301690 IC50 = 10000 nM T30082 CC3U6H 44301705 IC50 > 10000 nM T30082 C0G6UP 44301707 IC50 = 1300 nM T30082 C6W4ZF 44301727 IC50 = 3000 nM T30082 CUP5C9 44301796 IC50 = 1000 nM T30082 CT2A6Q 44303201 IC50 = 10000 nM T30082 C8S5AC 44305794 IC50 = 700 nM T30082 CM7IR4 44305795 IC50 = 380 nM T30082 C3NX2A 44305798 IC50 = 60 nM T30082 CL12EY 44305802 IC50 = 930 nM T30082 C5VI6E 44305803 IC50 = 3800 nM T30082 C8KGJ6 44305895 IC50 = 7600 nM T30082 C8LZ1B 44305960 IC50 = 21000 nM T30082 CTF46L 44306044 IC50 = 70 nM T30082 C5IS3D 44314031 IC50 = 23000 nM T30082 C9H4RO 44319895 IC50 = 53 nM T30082 CD5GZ9 44319908 IC50 = 10000 nM T30082 C0KQV9 44319925 IC50 = 19580 nM T30082 CL84KW 44319927 IC50 = 750 nM T30082 C4N5WR 44319929 IC50 = 90 nM T30082 C5QO8L 44319931 IC50 = 32 nM T30082 CZS05I 44319933 IC50 = 54 nM T30082 C92CKW 44319947 IC50 = 2670 nM T30082 C3XQ7C 44320086 EC50 = 100 nM T30082 CYB53A 44320110 IC50 < 500 nM T30082 C0I9EP 44320112 EC50 > 10000 nM T30082 CJ2W3N 44320122 EC50 = 2700 nM T30082 C82VSC 44320131 IC50 = 520 nM T30082 C1ZU8P 44320133 IC50 = 40 nM T30082 C3WA0S 44320152 IC50 = 43 nM T30082 CTVQ21 44320157 IC50 = 120 nM T30082 C3TR5O 44320163 IC50 = 540 nM T30082 CBNQ61 44320183 IC50 = 110 nM T30082 CJ3DB5 44320185 IC50 = 2570 nM T30082 C1DH8B 44320187 IC50 = 280 nM T30082 CDU1Z8 44320196 IC50 = 120 nM T30082 C2V6GW 44320240 EC50 = 2500 nM T30082 C96DMZ 44320295 EC50 = 1440 nM T30082 CZB9R1 44320296 EC50 = 890 nM T30082 C5HGT0 44320342 IC50 = 100 nM T30082 CNX78U 44320345 IC50 = 110 nM T30082 CMRK92 44320358 EC50 = 6600 nM T30082 CK8N9L 44320376 IC50 ~ 500 nM T30082 CTGW68 44320380 EC50 = 1880 nM T30082 C2I7MP 44320381 IC50 = 8 nM T30082 CED1Y7 44320382 EC50 = 43500 nM T30082 CAYD70 44320394 IC50 = 1000 nM T30082 C1FGB2 44320525 IC50 > 1000 nM T30082 C51CRA 44320527 IC50 = 79 nM T30082 CXA47P 44320541 IC50 = 390 nM T30082 CR2V1Q 44320543 IC50 = 41.5 nM T30082 C6YHJ4 44320549 IC50 = 50 nM T30082 CLG35I 44320569 Ki = 138.04 nM T30082 CU7H8Z 44320583 IC50 = 17 nM T30082 C20UNT 44320609 IC50 = 7 nM T30082 CH0U9R 44320631 EC50 = 290 nM T30082 CC6O8F 44320632 IC50 = 28 nM T30082 C0FZ2B 44320942 IC50 = 245000 nM T30082 CH3NS9 44321797 IC50 = 18580 nM T30082 C67ZKS 44325347 IC50 = 210 nM T30082 C6RS8G 44333218 IC50 = 406000 nM T30082 C0F3LH 44340178 IC50 = 104712.85 nM T30082 C8ZNT6 44340235 IC50 = 15848.93 nM T30082 CF4V0R 44340535 IC50 = 6165.95 nM T30082 C1OS3X 44341772 IC50 = 240.6 nM T30082 C0XI2G 44344490 IC50 = 110000 nM T30082 CA95RW 44344802 IC50 = 47000 nM T30082 CT1Q3S 44347198 IC50 = 760 nM T30082 CPXK27 44347214 IC50 = 10 nM T30082 CNY9B1 44347584 IC50 = 24 nM T30082 CVL5Y1 44347602 IC50 = 10 nM T30082 C7ABL6 44347792 IC50 > 100000 nM T30082 C31XIP 44354060 IC50 = 313 nM T30082 CB6E3P 44354097 IC50 = 606 nM T30082 C25JFX 44354109 IC50 = 150 nM T30082 C09POI 44357647 IC50 = 345143.74 nM T30082 C9TPB7 44357654 IC50 = 5970.35 nM T30082 CK63TC 44357655 IC50 = 5333.35 nM T30082 C8I5PJ 44357666 IC50 = 69023.98 nM T30082 C8IU7V 44357667 IC50 = 753355.56 nM T30082 CHUD79 44357680 IC50 = 3767.04 nM T30082 CIQG85 44357700 IC50 = 659.17 nM T30082 CO36AH 44357703 IC50 = 1798.87 nM T30082 CLO21E 44357712 IC50 = 238781.13 nM T30082 C73WOL 44357731 IC50 = 40831.94 nM T30082 CN6M5I 44357738 IC50 = 109.9 nM T30082 CD5Z7I 44357752 IC50 = 122461.62 nM T30082 CYZ6O9 44357806 IC50 = 1698.24 nM T30082 CV1QX7 44357818 IC50 = 33.96 nM T30082 CGXR18 44357831 IC50 = 152.05 nM T30082 C1A6MP 44357837 IC50 = 460 nM T30082 CM98SV 44357881 IC50 = 19952.62 nM T30082 CM8D3A 44357884 IC50 = 35000 nM T30082 C6XZ4O 44357902 IC50 = 39994.47 nM T30082 CTF92Z 44357904 IC50 = 6295.06 nM T30082 CC1N3T 44357916 IC50 = 3828247.43 nM T30082 CU4Q2V 44357985 IC50 = 1761976.05 nM T30082 CEJ9F2 44357987 IC50 = 11587773.56 nM T30082 C3P1TN 44357988 IC50 = 8128305.16 nM T30082 C1J0SR 44358056 IC50 = 3706807.22 nM T30082 CCY9M7 44358057 IC50 = 1729816.36 nM T30082 CXD43V 44358068 IC50 = 7079.46 nM T30082 C4H8OA 44358095 IC50 = 6165.95 nM T30082 C4UZC2 44358097 IC50 = 690239.8 nM T30082 C05RBY 44358110 IC50 = 5754.4 nM T30082 CRC09U 44358121 IC50 = 50118.72 nM T30082 C3OPV1 44358179 IC50 = 69183.1 nM T30082 CLP56M 44358199 IC50 = 33113.11 nM T30082 CQ7TC1 44358210 IC50 = 42657.95 nM T30082 CM9VG2 44358214 IC50 = 70794.58 nM T30082 C5GYN9 44358266 IC50 = 50118.72 nM T30082 COP8B7 44358267 IC50 = 13803.84 nM T30082 C6LO3N 44358273 IC50 = 5248.07 nM T30082 CY9MW4 44358283 IC50 = 6456.54 nM T30082 CC79ZF 44361495 IC50 = 2.2 nM T30082 CK6QX1 44361516 IC50 = 11.7 nM T30082 CGHX23 44361622 IC50 = 4.96 nM T30082 C3OHM0 44361641 IC50 = 1.76 nM T30082 CF4GR3 44361719 IC50 = 1.39 nM T30082 C0SZQ9 44362025 IC50 = 436 nM T30082 CF3H1M 44362158 IC50 = 76.9 nM T30082 C0YMK5 44364677 IC50 = 33000 nM T30082 CQU4V5 44366070 IC50 = 1800 nM T30082 CE7RW5 44366101 IC50 = 52400 nM T30082 C3EKJ1 44366110 IC50 = 3940 nM T30082 C84FRK 44369395 IC50 > 100000 nM T30082 CLZK10 44369408 IC50 > 100000 nM T30082 C3D9TR 44370789 IC50 = 3 nM T30082 C52LPH 44371758 IC50 = 230 nM T30082 C9LZ3A 44371762 IC50 = 3360 nM T30082 CS6Y9L 44371770 IC50 = 180 nM T30082 C9S8PR 44371772 IC50 = 160 nM T30082 CW2O7E 44371784 IC50 = 3840 nM T30082 COX76Y 44371839 IC50 = 160 nM T30082 CB6L5H 44371855 IC50 = 140 nM T30082 C7X0ZU 44371902 IC50 = 60 nM T30082 C81QMK 44371903 IC50 = 3170 nM T30082 CYPL76 44371904 IC50 = 4190 nM T30082 CY5E0V 44371918 IC50 = 670 nM T30082 CI25TC 44371926 IC50 = 5680 nM T30082 CPZ38Y 44372077 IC50 = 230 nM T30082 CTB8G1 44376824 IC50 = 1300 nM T30082 CE75QO 44376983 IC50 = 270000 nM T30082 CQKO52 44377194 IC50 = 440000 nM T30082 CH2DU4 44381982 IC50 = 42.2 nM T30082 CD8W7K 44381983 IC50 = 84.3 nM T30082 C39BIX 44385143 IC50 = 72.44 nM T30082 C57WPN 44388351 IC50 = 3860 nM T30082 CU6Q3K 44390121 Ki = 208.77 nM T30082 CJQ40I 44390138 Ki = 399.71 nM T30082 CO2C1T 44390186 Ki = 1004 nM T30082 CK7IW0 44390223 Ki = 1340 nM T30082 CS5JE9 44390234 Ki = 1590 nM T30082 CSW6Q0 44390235 Ki = 543.47 nM T30082 C0KH5F 44390238 Ki = 1330 nM T30082 CY4M9P 44390241 Ki = 62.06 nM T30082 C7X6JR 44390244 Ki = 865.03 nM T30082 CY3K5C 44390255 Ki = 505.09 nM T30082 C17QVZ 44390271 Ki = 514.05 nM T30082 CS4TL0 44390273 Ki = 266.41 nM T30082 C91YNH 44390278 Ki = 69.46 nM T30082 C9BE8H 44390283 Ki = 793.14 nM T30082 CDVT68 44390293 Ki = 77.66 nM T30082 C6RYB0 44390301 Ki = 403.05 nM T30082 C8LWJ6 44390309 Ki = 38.18 nM T30082 CVR3N5 44390334 Ki = 402.85 nM T30082 C9WKX0 44390337 Ki = 106.26 nM T30082 CALW31 44390341 Ki = 118.04 nM T30082 C2MJ0F 44390349 Ki = 217.13 nM T30082 C0Z6BU 44390361 Ki = 137.63 nM T30082 CW2XR7 44390392 Ki = 227.94 nM T30082 CW09ZP 44391786 IC50 = 230 nM T30082 CPZ3Y1 44391798 IC50 = 90 nM T30082 C8XH3P 44391811 IC50 = 60 nM T30082 C46ESP 44391828 IC50 = 420 nM T30082 C56SXM 44391858 Ki = 2300 nM T30082 C4XDV0 44392388 Ki = 1400 nM T30082 CW16VH 44392399 Ki = 360 nM T30082 CEC09G 44392415 Ki = 360 nM T30082 CP10BD 44392425 Ki = 250 nM T30082 C8SZ7C 44392426 Ki = 150 nM T30082 CE59SW 44392437 Ki = 160 nM T30082 CF7R5N 44392446 Ki = 160 nM T30082 C5PHC4 44392449 Ki = 170 nM T30082 CE9AS1 44392487 Ki = 200 nM T30082 CH0PM4 44392488 Ki = 300 nM T30082 CFUX63 44392498 Ki = 200 nM T30082 CQ5YC6 44392500 Ki = 130 nM T30082 C0F8YB 44393119 IC50 = 363.08 nM T30082 C5K3CW 44396585 IC50 = 8500 nM T30082 CDKL61 44396613 Ki = 5.754 nM T30082 CXSN45 44396628 Ki = 42.66 nM T30082 C0ER5W 44396629 IC50 = 120 nM T30082 CB4Y7H 44396640 Ki = 39.81 nM T30082 C6QE8M 44396641 IC50 = 7 nM T30082 C15VWH 44396642 IC50 = 6 nM T30082 C4CE2A 44396643 Ki = 4.571 nM T30082 CO94XT 44396651 IC50 = 750 nM T30082 CYF70Q 44396652 IC50 = 30000 nM T30082 CJ8E0D 44396653 Ki = 239.88 nM T30082 CILV80 44396690 IC50 = 250 nM T30082 CVOP24 44396691 Ki = 7.943 nM T30082 CIR4X6 44396692 Ki = 109.65 nM T30082 CUK27T 44396699 Ki = 1000 nM T30082 CNTL16 44396700 IC50 = 2570 nM T30082 CX8IH9 44396707 IC50 = 6.27 nM T30082 CTU61G 44396708 Ki = 109.65 nM T30082 C5S0OU 44396709 IC50 = 30 nM T30082 CC48EF 44396719 Ki = 89.13 nM T30082 COUB19 44396741 IC50 = 520 nM T30082 CG04OR 44396742 Ki = 19498.45 nM T30082 CUPM16 44396760 Ki = 0.4786 nM T30082 COV64Z 44396761 IC50 = 380 nM T30082 CY3V6K 44396774 Ki = 2.57 nM T30082 CO65ID 44396775 Ki = 53.7 nM T30082 C03OUX 44396801 Ki = 389.05 nM T30082 C4Y8EU 44396802 Ki = 1000 nM T30082 CYQI97 44396850 IC50 = 2670 nM T30082 CQLJ82 44396851 Ki = 52.48 nM T30082 C8P4KE 44396852 IC50 = 79 nM T30082 CHC6J3 44396856 Ki = 338.84 nM T30082 CR9U5A 44396900 IC50 = 28 nM T30082 C7OJY0 44396906 Ki = 891.25 nM T30082 C1HCB2 44396916 IC50 = 280 nM T30082 CWA7H5 44396917 IC50 = 190 nM T30082 CNBR80 44398165 IC50 = 17.3 nM T30082 C5P4KS 44398279 IC50 = 20.3 nM T30082 CX01VE 44398294 IC50 = 420 nM T30082 CN6PS1 44398377 IC50 = 8.11 nM T30082 C1M3ZD 44398397 IC50 = 1870 nM T30082 C2B5HS 44398438 IC50 = 393 nM T30082 C7IRF1 44398566 IC50 = 2090 nM T30082 CO2K3G 44399793 IC50 = 20000 nM T30082 CSQ5I6 44399806 IC50 = 20000 nM T30082 CPQ39J 44399838 IC50 = 20000 nM T30082 C04OBZ 44399845 IC50 = 20000 nM T30082 C1N0GH 44399869 IC50 = 20000 nM T30082 C7UQ8M 44399881 IC50 = 20000 nM T30082 CLJ3W7 44399942 IC50 = 20000 nM T30082 C4PI5D 44402368 IC50 = 32 ug.mL-1 T30082 CIG41P 44402369 IC50 = 137000 nM T30082 CG34OE 44402435 IC50 = 40.7 ug.mL-1 T30082 CQ0W4K 44402478 IC50 = 50 ug.mL-1 T30082 C76LZX 44402502 IC50 = 30 ug.mL-1 T30082 CB7O4H 44402580 IC50 = 35 ug.mL-1 T30082 C90XAH 44402596 IC50 = 15 ug.mL-1 T30082 CMF05N 44409456 IC50 = 82 nM T30082 CJ35GS 44409574 IC50 = 94 nM T30082 CP04JE 44410039 IC50 = 6940 nM T30082 C9ZHL5 44412131 Ki = 16.5 nM T30082 CQ12BX 44412132 Ki = 15.7 nM T30082 CHO3A1 44412135 Ki = 6.4 nM T30082 C4KN6X 44412186 Ki = 0.026 nM T30082 CAE21M 44413731 IC50 > 3000 nM T30082 C9U1ZG 44413802 IC50 > 5000 nM T30082 C90RTX 44413815 IC50 > 3000 nM T30082 CS32BR 44414004 IC50 = 284.2 nM T30082 C0YW2U 44414005 IC50 = 126.3 nM T30082 CLJ2Q6 44414008 IC50 = 3203.7 nM T30082 CQ27HV 44414014 IC50 = 1341.7 nM T30082 CUC68M 44414019 IC50 = 1012.9 nM T30082 C6F4WZ 44414020 IC50 = 73.6 nM T30082 CF0XV9 44417532 IC50 = 98 nM T30082 C98SME 44417548 IC50 = 40.5 nM T30082 CV7XP1 44417560 IC50 = 225 nM T30082 C0JYP1 44418744 IC50 = 5.08 nM T30082 C80MLQ 44418787 IC50 = 227 nM T30082 CG41JA 44419699 IC50 > 10000 nM T30082 CY8RQ9 44419966 IC50 > 10000 nM T30082 CXZ52T 44419971 IC50 > 10000 nM T30082 C7SN0Z 44421297 Ki = 104 nM T30082 C9I7EY 44421298 Ki = 12.2 nM T30082 CD3SJ4 44421300 IC50 = 3.311 nM T30082 CJ47UB 44421301 IC50 = 7.413 nM T30082 C8GY2A 44421302 IC50 = 6.607 nM T30082 CC64OM 44421303 IC50 = 36.31 nM T30082 CV7RQ4 44421304 IC50 = 63.1 nM T30082 CQ8V9A 44421305 IC50 = 169.82 nM T30082 CV46OY 44421933 IC50 = 594000 nM T30082 CHQ74U 44421934 IC50 = 1050000 nM T30082 CM2PQ9 44421939 IC50 = 565000 nM T30082 CPM30V 44421940 IC50 = 413000 nM T30082 CX7T8G 44421945 IC50 = 138000 nM T30082 CGN9K0 44421946 IC50 = 127000 nM T30082 CR4K2Y 44421950 IC50 = 155000 nM T30082 CF0SC4 44421951 IC50 = 3150 nM T30082 CH9WV0 44421967 IC50 = 7840 nM T30082 CQ6ZY2 44421972 IC50 = 2320 nM T30082 C4AF3S 44421973 IC50 = 3400 nM T30082 CO97PS 44421976 IC50 = 2180 nM T30082 C1SK6X 44421982 IC50 = 40000 nM T30082 C9FZP5 44421986 IC50 = 360000 nM T30082 CTD13B 44421991 IC50 = 433000 nM T30082 CCB15K 44423472 IC50 = 31000 nM T30082 CEQ6U7 44423479 IC50 = 1 nM T30082 C1P3IO 44424523 IC50 = 27900 nM T30082 CO9LC6 44427467 IC50 = 202 nM T30082 CM6GB7 44427468 IC50 = 2290 nM T30082 CEVO25 44427469 IC50 = 892 nM T30082 CJ64GU 44427470 IC50 = 303 nM T30082 CZ83QC 44427471 IC50 = 163 nM T30082 CPM03B 44427472 IC50 = 987 nM T30082 CCJH84 44427473 IC50 = 368 nM T30082 CN5CJ2 44427474 IC50 = 24600 nM T30082 CHQ62N 44427475 IC50 = 366 nM T30082 C6WDH3 44427476 IC50 = 122 nM T30082 CZTU76 44427477 IC50 = 310 nM T30082 CO1NJ5 44427478 IC50 = 62.1 nM T30082 CQ5G6X 44427479 IC50 = 714 nM T30082 C4M7RQ 44427480 IC50 = 2260 nM T30082 CLS78U 44427481 IC50 = 49.3 nM T30082 C5O1RW 44427482 IC50 = 148 nM T30082 C0AM6W 44427483 IC50 = 281 nM T30082 CE09QX 44427485 IC50 = 30300 nM T30082 CFMN40 44427486 IC50 = 1230 nM T30082 CS3AX5 44427487 IC50 = 2020 nM T30082 C9XM2E 44427488 IC50 = 1590 nM T30082 C0WMB1 44427489 IC50 = 2270 nM T30082 CPM76T 44427490 IC50 = 3100 nM T30082 CQ87RG 44427491 IC50 = 18100 nM T30082 CT38CX 44427492 IC50 = 80500 nM T30082 CSO3M0 44427493 IC50 = 10.5 nM T30082 CDE8A1 44428745 IC50 = 1288.25 nM T30082 C0C2DX 44428836 Ki > 100000 nM T30082 CZS9U1 44428842 Ki > 100000 nM T30082 CWR3Y1 44428843 Ki > 100000 nM T30082 CUT0H7 44428844 Ki > 100000 nM T30082 C0NHI2 44435121 IC50 > 50000 nM T30082 CIW9A7 44435348 IC50 = 299 nM T30082 C83BXH 44435798 Ki > 100000 nM T30082 C2VL9X 44436444 IC50 = 82.5 nM T30082 CS37XC 44436445 IC50 = 135.4 nM T30082 CP40RO 44436447 IC50 = 230.8 nM T30082 COU3R7 44436448 IC50 = 231.5 nM T30082 C28MNB 44436451 IC50 = 286.4 nM T30082 C4WI8J 44436452 IC50 = 383.5 nM T30082 CPO17N 44445157 IC50 = 182 nM T30082 CBE50J 44445172 IC50 = 12022.64 nM T30082 CW4E8M 44445173 IC50 = 20892.96 nM T30082 C2OPV6 44445174 IC50 = 13803.84 nM T30082 C2OT6L 44445175 IC50 = 8912.51 nM T30082 CMH2X0 44445176 IC50 = 1202.26 nM T30082 C9TPF3 44445177 IC50 = 1288.25 nM T30082 CO6LF2 44445178 IC50 = 5370.32 nM T30082 CG68ZA 44445179 IC50 = 1288.25 nM T30082 C7TYD4 44445180 IC50 = 933.25 nM T30082 CY5Z8M 44445181 IC50 = 6456.54 nM T30082 CIFZ16 44445182 IC50 = 1202.26 nM T30082 CDAL58 44445183 IC50 = 8128.31 nM T30082 C8Y7CU 44445184 IC50 = 1412.54 nM T30082 CN7H8M 44445185 IC50 = 5128.61 nM T30082 C2D4FR 44445841 IC50 = 9010 nM T30082 CF9SH8 44446101 Ki = 313700 nM T30082 C5K6XG 44446102 Ki = 159000 nM T30082 C7IH4Y 44446104 Ki = 150900 nM T30082 CE7M5J 44446106 Ki = 115900 nM T30082 CIQ4O9 44446113 Ki = 140200 nM T30082 CX9K6E 44447995 IC50 = 952 nM T30082 CI1XD0 44448000 IC50 = 43900 nM T30082 CXP2J1 44451644 IC50 = 1100 nM T30082 CZUW95 44455900 IC50 = 551 nM T30082 CC1M7L 44455901 IC50 = 2770 nM T30082 CIQ06V 44456429 IC50 = 4570 nM T30082 CV0A2R 44456430 IC50 = 327 nM T30082 CKN04W 44456431 IC50 = 4230 nM T30082 CYVS69 44456474 IC50 = 267000 nM T30082 CINB34 44456475 IC50 = 181 nM T30082 C5L8AQ 44545550 IC50 = 659 nM T30082 C02WLM 44545753 IC50 = 1213 nM T30082 CXY10R 44545757 IC50 = 333 nM T30082 COY01J 44545824 IC50 = 13300 nM T30082 C86IVN 44545828 IC50 = 135 nM T30082 CRWT79 44545901 IC50 = 18 nM T30082 C96YPZ 44546167 IC50 = 259 nM T30082 CS5OI0 44546169 IC50 = 18 nM T30082 CZH21K 44546426 IC50 = 496 nM T30082 CATK49 44546490 IC50 = 1037 nM T30082 COZ20N 44546493 IC50 = 493 nM T30082 CJ41TE 44550606 IC50 = 950 nM T30082 CTYA64 44550607 IC50 = 250 nM T30082 CP0O8Q 44550608 IC50 = 100 nM T30082 CPWV46 44550725 IC50 = 530 nM T30082 CQV8G2 44550726 IC50 = 500 nM T30082 CNP4T9 44550727 IC50 = 180 nM T30082 CPT1O4 44550728 IC50 = 270 nM T30082 CLFZ14 44550729 IC50 = 440 nM T30082 CLVX32 44550849 IC50 = 300 nM T30082 CIT5G7 44561891 IC50 > 100000 nM T30082 C90BGR 44561892 IC50 > 100000 nM T30082 C9RGX4 44561893 IC50 > 100000 nM T30082 CU7NP5 44561930 IC50 > 100000 nM T30082 CV21IQ 44561931 IC50 > 100000 nM T30082 CR08WA 44561932 IC50 > 100000 nM T30082 C0G3SJ 44580530 Ki = 6320 nM T30082 C1AO5C 44580576 Ki = 11190 nM T30082 C9G1VW 44580577 Ki = 4130 nM T30082 C5G2VP 44580578 Ki = 1908 nM T30082 CP4FT6 44580579 Ki = 2214 nM T30082 C6PLC4 44580639 Ki = 3330 nM T30082 CB1ZL8 44580640 Ki = 7970 nM T30082 CQ6U4X 44580641 Ki = 34030 nM T30082 CL73ZJ 44580642 Ki = 130 nM T30082 CK4M5S 44580643 Ki = 280 nM T30082 C8N4ZQ 44580644 Ki = 15.4 nM T30082 CMR90Y 44580645 Ki = 6.21 nM T30082 CWHP70 44580646 Ki = 6.75 nM T30082 CGJ3O4 44586009 IC50 = 8.32 nM T30082 CRJC18 44587246 IC50 = 22100 nM T30082 CM27UT 44587247 IC50 = 9900 nM T30082 CP4G7M 44587346 IC50 = 18800 nM T30082 CL68VX 44587347 IC50 = 70600 nM T30082 C37PVZ 44587494 IC50 = 71100 nM T30082 CMP67W 44587524 IC50 = 49400 nM T30082 CGK71P 44587544 IC50 = 5900 nM T30082 CIF0E9 44587921 IC50 = 40000 nM T30082 C7MW1Z 44589810 IC50 = 5470 nM T30082 CL1PQ6 44604353 IC50 > 30000 nM T30082 C34RFE 44604423 IC50 > 30000 nM T30082 C6K8GE 45049498 IC50 = 36000 nM T30082 CTBO39 45130737 IC50 = 636000 nM T30082 CJP71Z 45261769 IC50 = 24.7 nM T30082 C2MN6D 45261778 IC50 = 5.4 nM T30082 CTYU71 45261781 IC50 = 21.8 nM T30082 CY6GX3 45261793 IC50 = 210 nM T30082 CZ16LQ 45261805 IC50 = 82.6 nM T30082 C67KQI 45261809 IC50 = 11.7 nM T30082 CW09OL 45261830 IC50 = 0.32 nM T30082 C1PJ0D 45262383 IC50 = 10500 nM T30082 C9XE1W 45262387 IC50 = 45800 nM T30082 CZE2Q8 45262393 IC50 = 41200 nM T30082 CKG50Z 45262394 IC50 = 550 nM T30082 CI16EA 45262395 IC50 = 300 nM T30082 CK2W6S 45262399 IC50 = 530 nM T30082 CS6LQ1 45262424 IC50 = 7000 nM T30082 CHMC90 45262425 IC50 = 15700 nM T30082 C56PRD 45262427 IC50 = 19000 nM T30082 CM6PI0 45262428 IC50 = 760 nM T30082 CP24DI 45262431 IC50 > 1300000 nM T30082 C63JWM 45262432 IC50 = 17900 nM T30082 CFP2A4 45262433 IC50 >> 1000000 nM T30082 CL46NA 45262434 IC50 = 17900 nM T30082 CWP3B7 45262437 IC50 = 13700 nM T30082 COP32V 45262453 IC50 = 1480 nM T30082 C7PU8O 45262463 IC50 = 9 nM T30082 CLJV07 45262466 IC50 = 2900 nM T30082 C3T6CD 45262469 IC50 = 25500 nM T30082 C5L8EQ 45262470 IC50 >> 1000000 nM T30082 C23-FEB 45262473 IC50 = 3960 nM T30082 CL8OE1 45262474 IC50 = 26 nM T30082 CS4BV6 45262475 IC50 = 13 nM T30082 CVZ12D 45262477 IC50 = 1070 nM T30082 CY3LZ0 45262481 IC50 = 14600 nM T30082 C7EFJ5 45262486 IC50 = 2150 nM T30082 CCG3F5 45262487 IC50 = 24500 nM T30082 CJB7K6 45262489 IC50 = 38600 nM T30082 CB8TJ3 45262490 IC50 = 1780 nM T30082 CLY83X 45262491 IC50 > 500000 nM T30082 C7NI9X 45262500 IC50 = 860 nM T30082 CBN47U 45262501 IC50 = 53 nM T30082 CS89CF 45262502 IC50 = 14900 nM T30082 C0P2BE 45262503 IC50 = 17700 nM T30082 C3IDO6 45262507 IC50 = 7300 nM T30082 CD2QW6 45262508 IC50 = 2150 nM T30082 CY17RU 45263524 IC50 = 170 nM T30082 CGE36P 45265144 IC50 = 12.4 nM T30082 CH6SJ9 45265175 IC50 = 6.8 nM T30082 CHA28P 45265179 IC50 = 79.6 nM T30082 CW0XO4 45265314 IC50 = 2500 nM T30082 C2SA5R 45265370 IC50 = 72400 nM T30082 CYGK37 45265574 IC50 = 439000 nM T30082 CRX07O 45265577 IC50 > 500000 nM T30082 C3XS2M 45265585 IC50 = 11300 nM T30082 C5QY1I 45265587 IC50 = 460 nM T30082 CFRU23 45265609 IC50 = 510 nM T30082 CO57DP 45265613 IC50 = 3600 nM T30082 CJ9D0H 45265615 IC50 = 43900 nM T30082 COW2D8 45266157 IC50 = 100 nM T30082 CHE19F 45266158 IC50 = 200 nM T30082 CNJ5W8 45266159 IC50 = 180 nM T30082 C46BXK 45266162 IC50 = 34 nM T30082 CYVD61 45266173 IC50 = 5.44 nM T30082 CF80CX 45266174 IC50 = 6.75 nM T30082 COP92A 45266176 IC50 = 6.54 nM T30082 C1LOR7 45266221 IC50 = 125 nM T30082 CO9LU8 45266222 IC50 > 10000 nM T30082 CT01NJ 45267086 IC50 = 22800 nM T30082 C4HD1L 45269664 IC50 = 14500 nM T30082 CO4K0N 45269909 IC50 > 10000 nM T30082 C0NU9K 45481993 IC50 = 4780 nM T30082 CYG78R 45481994 IC50 = 6450 nM T30082 CT24FL 45481995 IC50 = 50000 nM T30082 C3GF6X 45481996 IC50 = 8.69 nM T30082 CQ4XH0 45481997 IC50 = 13.7 nM T30082 COH60K 45481998 IC50 = 8080 nM T30082 C3MAF0 45481999 IC50 = 50000 nM T30082 C9EU7D 45482000 IC50 = 27100 nM T30082 CMJ67D 45482002 IC50 = 3.95 nM T30082 C7SZX8 45482003 IC50 = 5.96 nM T30082 CZ1U4F 45482005 IC50 = 7690 nM T30082 C87IMV 45482006 IC50 = 7270 nM T30082 CJ0N1L 45482008 IC50 = 50000 nM T30082 C28EID 45482009 IC50 = 50000 nM T30082 C06QEF 45482010 IC50 = 2510 nM T30082 C6OAT0 45482011 IC50 = 14700 nM T30082 C1ZDB5 45482012 IC50 = 2920 nM T30082 CW3HA5 45482013 IC50 = 11700 nM T30082 CG94LO 45482014 IC50 = 22400 nM T30082 CF2RM5 45482015 IC50 = 19200 nM T30082 CBKZ29 45482016 IC50 = 9.66 nM T30082 CG3X5H 45482017 IC50 = 5100 nM T30082 C90UIA 45482018 IC50 = 43.3 nM T30082 CJW20I 45482019 IC50 = 810 nM T30082 CGW25K 45482020 IC50 = 855 nM T30082 CL91TN 45482021 IC50 = 664 nM T30082 CXQ0Y4 45486365 IC50 = 50 nM T30082 CQFC83 45488333 IC50 = 2400 nM T30082 CIG1O6 46211767 Ki = 3100 nM T30082 C4X9KL 46225676 IC50 = 1630 nM T30082 C9B2QT 46226577 IC50 = 31 nM T30082 C7GH1V 46226589 IC50 = 29 nM T30082 CJYE32 46226600 IC50 = 84 nM T30082 CV28SE 46226601 IC50 = 22 nM T30082 CG34XN 46226620 IC50 = 24 nM T30082 C76PFG 46226629 IC50 = 51 nM T30082 CY4TZ8 46226630 IC50 = 25 nM T30082 C1IT5R 46226643 IC50 = 40 nM T30082 CY6U7A 46226644 IC50 = 41 nM T30082 CBJ38C 46226649 IC50 = 31 nM T30082 C9B4QG 46226660 IC50 = 31 nM T30082 CC64KH 46227076 IC50 = 7 nM T30082 C1MSE9 46228657 IC50 = 1140 nM T30082 C31MLQ 46228658 IC50 = 28700 nM T30082 CT9CI3 46228685 IC50 = 630 nM T30082 CIK7S8 46228686 IC50 = 4930 nM T30082 C2V4QP 46228687 IC50 = 11700 nM T30082 CC85MY 46228688 IC50 = 2900 nM T30082 CE86KJ 46228721 IC50 = 1610 nM T30082 C7CY5S 46228722 IC50 = 3950 nM T30082 C7W8OG 46228723 IC50 = 1530 nM T30082 CK62AH 46228724 IC50 = 1320 nM T30082 C20GZR 46228760 IC50 = 890 nM T30082 C4O9CE 46228761 IC50 = 890 nM T30082 CLUW07 46228762 IC50 = 180 nM T30082 CJ5YZ9 46228787 IC50 = 190 nM T30082 CJ2D5H 46228788 IC50 = 200 nM T30082 CJG67U 46228789 IC50 = 380 nM T30082 CTBX50 46228809 IC50 = 510 nM T30082 C6O3FS 46228810 IC50 = 110 nM T30082 C0PHL3 46228811 IC50 = 5380 nM T30082 C9IE5S 46228812 IC50 = 180 nM T30082 C7POL5 46228839 IC50 = 56 nM T30082 C1E3LQ 46228840 IC50 = 52 nM T30082 CUE0H9 46229068 IC50 = 7000 nM T30082 CB6C1T 46229099 IC50 = 600000 nM T30082 C6QA8X 46229101 IC50 > 1000000 nM T30082 CEBO01 46229144 Ki = 810 nM T30082 C7Q6RX 46231880 IC50 = 25000 nM T30082 C0VIS5 46854881 IC50 = 5.5 nM T30082 CD0Q4G 46855034 IC50 = 0.5 nM T30082 C7L1OM 46861819 Ki = 24 nM T30082 CBO8D7 46863225 IC50 = 520 nM T30082 CJ16FO 46866088 Ki = 140 nM T30082 CI69YW 46867253 IC50 = 1900 nM T30082 C3U7VW 46867254 IC50 = 1000 nM T30082 CH5PS4 46867255 IC50 = 2000 nM T30082 CUMA45 46867256 IC50 = 1800 nM T30082 CQH53B 46867382 IC50 = 2100 nM T30082 CT19SR 46867383 IC50 = 2000 nM T30082 C13URS 46867384 IC50 = 1800 nM T30082 C2MSV7 46877440 IC50 = 4.5 nM T30082 C8SX4T 46877447 IC50 = 5116818.36 nM T30082 CZIT18 46877450 Ki = 4.467 nM T30082 C5I7EO 46877451 IC50 = 32 nM T30082 CX7J9D 46880263 IC50 = 2010000 nM T30082 CM6PJ3 46880264 IC50 = 1990000 nM T30082 C61VGD 46880266 IC50 = 2360000 nM T30082 C5G4FV 46880955 IC50 = 241000 nM T30082 CHNP43 46888221 IC50 = 25080 nM T30082 C5RJ8F 46889315 IC50 = 160 nM T30082 C91OJY 46889316 IC50 = 261 nM T30082 C73CLY 46889317 IC50 = 3700 nM T30082 C3VKL5 46889330 IC50 = 400 nM T30082 C7K3LC 46889331 IC50 = 750 nM T30082 C8WI5S 46889332 IC50 = 170 nM T30082 CY9GA8 46889333 IC50 = 1600 nM T30082 CQ7DW1 46889334 IC50 = 4800 nM T30082 C06YJV 46889354 IC50 = 54 nM T30082 CQS07A 46889355 IC50 = 170 nM T30082 C6IA5F 46889356 IC50 = 144100 nM T30082 C2DSK4 46889357 IC50 = 2.99 nM T30082 CE8I7V 46889391 IC50 = 1490 nM T30082 C4DN0E 46889392 IC50 = 0.52 nM T30082 CCT3P0 46889408 IC50 = 150 nM T30082 C57YJR 46889409 IC50 = 2100 nM T30082 C9JR8O 46889410 IC50 = 15000 nM T30082 CS96WZ 46889411 IC50 = 5.7 nM T30082 C9CUJ7 46889412 IC50 = 1.8 nM T30082 CUQ8F7 46889413 IC50 = 9.81 nM T30082 CXN7M3 46889414 IC50 = 4.94 nM T30082 C6UZH1 46889433 IC50 = 10000 nM T30082 C9LT7Q 46889434 IC50 = 300 nM T30082 C7DX6T 46889435 IC50 = 4400 nM T30082 C0Z2FH 46889436 IC50 = 0.02 nM T30082 CS02LM 46889437 IC50 = 0.06 nM T30082 CH7P9W 46889459 IC50 = 2.2 nM T30082 CM74LC 46889614 IC50 = 13000 nM T30082 C39IKO 46889615 IC50 = 100000 nM T30082 CA19WP 46889616 IC50 = 57000 nM T30082 C40XNS 46889617 IC50 = 54000 nM T30082 C9R0TX 46889618 IC50 = 60000 nM T30082 C27MEK 46889620 IC50 = 24.7 nM T30082 CP0SK6 46889649 IC50 = 12600 nM T30082 C7JA1M 46889651 IC50 = 1300 nM T30082 CQXF23 46889654 IC50 = 10000 nM T30082 C7V5MI 46889656 IC50 = 8100 nM T30082 C5V4SB 46889658 IC50 = 1200 nM T30082 CA24BQ 46889660 IC50 = 30 nM T30082 CAJ8B4 46889675 IC50 = 700 nM T30082 CA9MR5 46889677 IC50 = 24500 nM T30082 C4PTS0 46889679 IC50 = 200 nM T30082 CWS1M3 46889681 IC50 = 1350 nM T30082 C8PTW9 46889683 IC50 = 1100 nM T30082 C5XZA8 46889706 IC50 = 1600 nM T30082 CD1GW6 46889708 IC50 = 19500 nM T30082 C1ARO0 46889709 IC50 = 4000 nM T30082 C7QT3E 46889711 IC50 = 1100 nM T30082 CJ18FA 46889713 IC50 = 7100 nM T30082 CFL51J 46889714 IC50 = 24000 nM T30082 CZX27V 46889717 IC50 = 1.5 nM T30082 C4ADZ5 46889736 IC50 = 12600 nM T30082 CHEB93 46889738 IC50 = 33600 nM T30082 CLT3A2 46889740 IC50 = 20500 nM T30082 CQ6X0K 46889742 IC50 = 2500 nM T30082 CTJR65 46889744 IC50 = 350 nM T30082 CT91YH 46889746 IC50 = 99 nM T30082 CT76QE 46889747 IC50 = 120 nM T30082 C4HG2Z 46889748 IC50 = 100 nM T30082 C4QW2C 46889749 IC50 = 100 nM T30082 CN6GZ3 46889750 IC50 = 0.7 nM T30082 C6UX3V 46889751 IC50 = 3 nM T30082 CBC85E 46889778 IC50 = 4500 nM T30082 CT97NG 46889780 IC50 = 27000 nM T30082 CXN70S 46889782 IC50 = 9500 nM T30082 CJ5CM0 46889784 IC50 = 50000 nM T30082 CKQH41 46889785 IC50 = 8 nM T30082 CE2D4Q 46889786 IC50 = 114 nM T30082 CAOG01 46889787 IC50 = 10 nM T30082 CFT0U1 46889788 IC50 = 4000 nM T30082 C68NJW 46889830 IC50 = 90 nM T30082 CRDG78 46889831 IC50 = 154 nM T30082 CO6M2H 46889832 IC50 = 42 nM T30082 C1K8QP 46889860 IC50 = 68 nM T30082 CL93VH 46889861 IC50 = 1330 nM T30082 C3T7JR 46889862 IC50 = 69 nM T30082 CBN3F0 46889863 IC50 = 93 nM T30082 C8GPE1 46889864 IC50 = 62 nM T30082 C7GFW2 46889865 IC50 = 506 nM T30082 CD2R1O 46889866 IC50 = 13 nM T30082 CR58XB 46889867 IC50 = 250 nM T30082 CB83LV 46889868 IC50 = 2.5 nM T30082 CND35Z 46889869 IC50 = 13000 nM T30082 CR6JG7 46889896 IC50 = 21 nM T30082 CENZ67 46889897 IC50 = 68 nM T30082 C83ANR 46889898 IC50 = 1.49 nM T30082 CHR7C8 46889899 IC50 = 894 nM T30082 C04CYW 46891016 IC50 = 24900 nM T30082 C4JIH7 46891058 IC50 = 18400 nM T30082 C86UFR 46891061 IC50 = 26400 nM T30082 C5L9PR 46891062 IC50 = 20400 nM T30082 C9FAE8 46891063 IC50 = 8800 nM T30082 C5AYZ0 46891117 IC50 = 5500 nM T30082 CF5CQ7 46891118 IC50 = 14700 nM T30082 C20CPR 46891119 IC50 = 12800 nM T30082 CAB5N0 46891120 IC50 = 17500 nM T30082 CZQL62 46897981 IC50 = 25.4 nM T30082 C4TWY7 46897983 IC50 = 14.6 nM T30082 CDG49K 46897985 IC50 = 145 nM T30082 CA7CK3 46897987 IC50 = 300 nM T30082 CO1PS9 46905531 IC50 = 1698.24 nM T30082 CQ57HG 46905532 IC50 = 501.19 nM T30082 C3I0GL 46905533 IC50 = 3715.35 nM T30082 C07AOG 46905534 IC50 = 1513.56 nM T30082 C7T2GX 46909057 IC50 = 1630 nM T30082 C3QW2P 46933840 Ki = 540 nM T30082 CY7ZW5 46937311 IC50 = 3.61 nM T30082 CXJ04C 49796971 IC50 = 100 nM T30082 CJH50R 49797481 IC50 > 100000 nM T30082 CC86IT 49799305 IC50 = 26.1 nM T30082 C4FHO0 49845187 IC50 = 9550000 nM T30082 CA9E5S 49845368 IC50 = 18620000 nM T30082 C6SE1Z 49845372 IC50 = 1950000 nM T30082 C6BC2U 49845373 IC50 = 5490000 nM T30082 C7IJ3C 49857726 Ki > 100000 nM T30082 C04NYX 49857906 Ki > 100000 nM T30082 CDT4Y6 49857907 Ki > 100000 nM T30082 C5XS3G 49857908 Ki > 100000 nM T30082 CHRB62 49857909 Ki > 100000 nM T30082 CV7J6X 49857910 Ki > 100000 nM T30082 CYU39N 49857911 Ki > 100000 nM T30082 C5WZL0 49857912 Ki > 100000 nM T30082 CCG80U 49858100 Ki > 100000 nM T30082 CCN05H 49858101 Ki > 100000 nM T30082 C7IP6N 49861304 IC50 = 1480000 nM T30082 CGP6T3 49864504 Ki = 390 nM T30082 CVI76Z 49864528 Ki = 970 nM T30082 C29TIX 50896785 IC50 = 9780 nM T30082 CT8MQ7 50908834 IC50 = 58200 nM T30082 CTQX80 50942800 IC50 = 12 nM T30082 C8DS0J 50942802 IC50 = 5 nM T30082 CA43KF 51026481 IC50 = 321 nM T30082 C9VXK3 51039357 IC50 = 7000 nM T30082 CU36CR 51039359 IC50 = 17000 nM T30082 C8X5WJ 51039361 IC50 = 250000 nM T30082 C1BA7H 51039363 IC50 = 8000 nM T30082 C4RQZ0 51039365 IC50 = 300 nM T30082 C61UMV 51042596 IC50 = 2000 nM T30082 CDP03R 51076628 Ki = 0.0056 nM T30082 C2I3RA 51346780 IC50 = 50 nM T30082 C4MH6G 51346832 IC50 = 5 nM T30082 C9AZ3J 51357040 IC50 > 10000 nM T30082 C8T1BE 51357043 IC50 = 8200 nM T30082 C3BRM2 51357044 IC50 = 6300 nM T30082 CIZ96K 51357316 IC50 = 4200 nM T30082 C5RXF2 51357319 IC50 > 10000 nM T30082 C6G9SM 51357595 IC50 > 25000 nM T30082 C1R0DP 51357597 IC50 > 10000 nM T30082 CU0I5S 51357598 IC50 > 10000 nM T30082 CE3H6X 51357599 IC50 > 10000 nM T30082 CGV79B 51357600 IC50 = 9700 nM T30082 C6S1KB 51357868 IC50 = 8600 nM T30082 C7QPU6 52110752 IC50 = 6600 nM T30082 CD52WQ 52111959 IC50 = 8600 nM T30082 CEGS83 52940502 IC50 = 39 nM T30082 CFCN62 52940766 IC50 = 32 nM T30082 CJKY93 52940773 IC50 = 41130 nM T30082 C5PJL4 52940842 IC50 = 66000 nM T30082 CLD3A0 52941194 IC50 = 5120 nM T30082 CN8XA0 52941218 IC50 = 7300 nM T30082 C9M1WZ 52941440 IC50 = 3120 nM T30082 CGUC34 52941525 IC50 = 11200 nM T30082 CRN6L2 52941538 IC50 = 8600 nM T30082 CS0EM5 52941653 IC50 = 14300 nM T30082 C8GBU1 52942019 IC50 = 330 nM T30082 CO0T9J 52942129 IC50 = 15370 nM T30082 CH72NB 52942352 IC50 = 7600 nM T30082 CNV97A 52943312 IC50 = 9860 nM T30082 C5ZMT7 52943313 IC50 = 8260 nM T30082 C5REL0 52944408 IC50 = 245.3 nM T30082 CX3QB9 52944508 IC50 = 6100 nM T30082 CFW1C4 52944509 IC50 = 3700 nM T30082 C7SP1X 52944510 IC50 = 4200 nM T30082 C8QAK5 52944789 IC50 = 6860 nM T30082 C1YE4K 52945609 IC50 = 830 nM T30082 CQ9NW3 52945615 IC50 = 8.11 nM T30082 CDV49N 52945656 IC50 = 3560 nM T30082 CA7T6Q 52945658 IC50 = 17.3 nM T30082 C4T7LB 52946247 IC50 = 2120 nM T30082 CC3Y8J 52946329 IC50 = 3700 nM T30082 C3F7VC 52946604 IC50 = 74 nM T30082 CV0EI4 52946669 IC50 = 387.5 nM T30082 C4MUA3 52946981 IC50 = 5200 nM T30082 CUI0R5 52947430 IC50 = 46000 nM T30082 CB3Q5S 52947614 IC50 = 4200 nM T30082 CF73YD 52947766 IC50 = 4300 nM T30082 C31DGQ 52948031 IC50 = 40 nM T30082 CQRK41 52948055 IC50 = 21000 nM T30082 CNQ6I9 52948187 IC50 = 12200 nM T30082 C5EN7Q 52948540 IC50 = 7260 nM T30082 CL0H4F 52948833 IC50 = 6600 nM T30082 C3ORW4 52949034 IC50 = 66 nM T30082 CV1O6X 52949321 IC50 = 160.8 nM T30082 C5YZ4Q 52949858 IC50 = 100000 nM T30082 CZ9RC2 52949932 IC50 = 4200 nM T30082 CTNM64 52950058 IC50 = 13200 nM T30082 CN0D7O 52950125 IC50 = 4300 nM T30082 C8ZKR5 52952236 IC50 = 620 nM T30082 C4JG6W 52952244 IC50 = 62 nM T30082 CIO3V4 52952919 IC50 = 25 nM T30082 C61YEU 52952920 IC50 = 24 nM T30082 C9T8YE 52952921 IC50 = 210 nM T30082 CDYC75 52952922 IC50 = 257 nM T30082 C4Z6WM 52952958 IC50 = 68 nM T30082 CPMW48 53231243 IC50 = 130 nM T30082 CD4NP3 53231341 IC50 = 210 nM T30082 C6RE1G 53231342 IC50 = 550 nM T30082 CK64RX 53231343 IC50 = 720 nM T30082 C4VE2O 53231344 IC50 = 217 nM T30082 CNC2D0 53231345 IC50 = 107 nM T30082 C0Z3AM 53231442 IC50 = 144 nM T30082 C5A3YX 53231443 IC50 = 143 nM T30082 CPM56F 53231444 IC50 = 810 nM T30082 CO40KS 53231445 IC50 = 110 nM T30082 C5M0OA 53242257 Ki = 3100 nM T30082 CQY69D 53248755 IC50 = 12600 nM T30082 C9EL0U 53306553 IC50 > 10000 nM T30082 C3DS7L 53316786 IC50 = 19000 nM T30082 CM6D9A 53316924 IC50 = 8500 nM T30082 CR7D2M 53316925 IC50 = 22900 nM T30082 C4WJV0 53316929 IC50 = 125.89 nM T30082 CMO98A 53316982 IC50 = 0.4898 nM T30082 C39OMW 53316983 IC50 = 42.66 nM T30082 CSB3J2 53317474 IC50 = 14.13 nM T30082 CU9L1W 53318226 IC50 = 33.11 nM T30082 C4M5UX 53318264 IC50 = 52.48 nM T30082 C54XTQ 53318265 IC50 = 0.7943 nM T30082 C9HO1L 53319040 IC50 = 3000 nM T30082 C50KUO 53319583 IC50 = 14000 nM T30082 C3MW8L 53319585 IC50 = 346.74 nM T30082 C67YGU 53320725 IC50 = 37 nM T30082 CY9HE5 53320727 IC50 = 26 nM T30082 CF0AC4 53320729 IC50 = 3400 nM T30082 CY7J8V 53320731 IC50 = 300 nM T30082 CE3M5X 53320877 IC50 = 25800 nM T30082 CNZH62 53320880 IC50 = 1.288 nM T30082 C0DUN8 53321516 IC50 = 500 nM T30082 C69OQW 53321610 IC50 = 89.13 nM T30082 CFKJ51 53322024 IC50 = 24 nM T30082 CUR1C7 53322213 IC50 = 5.129 nM T30082 C8LI6S 53322214 IC50 = 4.898 nM T30082 C6CO4P 53322255 IC50 = 15.85 nM T30082 CH1O9A 53322846 IC50 = 13000 nM T30082 C26USF 53323382 IC50 = 16 nM T30082 CZT5X1 53323384 IC50 = 10000 nM T30082 C4W2QD 53323550 IC50 = 151.36 nM T30082 CJT42H 53323551 IC50 = 64.57 nM T30082 C0MY6W 53323596 IC50 = 2.884 nM T30082 C2RJQ1 53324171 IC50 = 446000 nM T30082 CE0W5F 53324336 IC50 = 700 nM T30082 CM1KA7 53324700 IC50 = 24000 nM T30082 C1XL0O 53324702 IC50 = 2000 nM T30082 C6YMK9 53324854 IC50 = 30200 nM T30082 C2V6HQ 53324855 IC50 = 29800 nM T30082 CPMX34 53324859 IC50 = 1.096 nM T30082 CV7IW2 53324894 IC50 = 4.571 nM T30082 C4YWN2 53326005 IC50 = 32 nM T30082 CC43BJ 53326130 IC50 = 2.512 nM T30082 CVI6L8 53326131 IC50 = 8.71 nM T30082 CW8ZV1 53326729 IC50 = 300 nM T30082 CK45JD 53361165 IC50 = 0.815 nM T30082 CTSC36 53361167 IC50 = 0.784 nM T30082 CIP6E3 53361169 IC50 = 0.809 nM T30082 CC65WR 53484185 IC50 = 8000 nM T30082 CZE6P3 53484186 IC50 = 10000 nM T30082 CWK2J9 54097201 IC50 = 41 nM T30082 CDCR53 54577393 IC50 = 13.9 nM T30082 CUSF85 54577394 Ki = 1.01 nM T30082 CVJA50 54577395 IC50 = 12.1 nM T30082 CXOH83 54577607 IC50 = 455 nM T30082 C6S8KE 54580363 IC50 = 25000 nM T30082 CM27VW 54580364 IC50 = 14200 nM T30082 CD8PN5 54580372 IC50 = 418000 nM T30082 CT2L8P 54580374 IC50 = 6000 nM T30082 C7DH8A 54580376 IC50 = 800 nM T30082 C1IE9P 54580388 IC50 = 20 nM T30082 C3ENI1 54580389 IC50 = 744 nM T30082 C0DW4J 54580410 IC50 = 21600 nM T30082 C2SK5X 54580955 IC50 = 11600 nM T30082 CN20LZ 54581356 IC50 = 3 nM T30082 C4XJ1D 54581366 IC50 = 18800 nM T30082 C6KVB5 54581375 IC50 = 80 nM T30082 CBH4L1 54581388 IC50 = 43 nM T30082 C9HWQ0 54581416 IC50 = 19900 nM T30082 C23NPW 54582394 IC50 = 9000 nM T30082 CH60OU 54582403 IC50 = 298 nM T30082 C1MZ0J 54582404 IC50 = 3003 nM T30082 CX8N5Y 54582406 IC50 = 618 nM T30082 C2DPX4 54582421 IC50 = 15300 nM T30082 CNR5O3 54582422 IC50 = 26400 nM T30082 C06NMW 54582423 IC50 = 20200 nM T30082 CRJ8S6 54582424 IC50 = 28800 nM T30082 CT3O9A 54583223 IC50 = 9 nM T30082 CXVQ08 54583385 IC50 = 76 nM T30082 C7WS9L 54583386 IC50 = 6 nM T30082 C8NXY5 54583387 IC50 = 25 nM T30082 C5TNU0 54583408 IC50 = 12400 nM T30082 C5XHR3 54583948 IC50 = 1800 nM T30082 C21PHC 54584309 IC50 = 14 nM T30082 CZ8E5U 54584310 IC50 = 9 nM T30082 CH7JX8 54584326 IC50 = 40000 nM T30082 CZW86O 54584337 IC50 = 159 nM T30082 CVB76W 54584338 IC50 = 7 nM T30082 CD2JE7 54584897 IC50 = 1200000 nM T30082 CW8EU4 54585277 IC50 = 11 nM T30082 C9VCF6 54585278 IC50 = 3 nM T30082 C6AZ5T 54585295 IC50 = 22900 nM T30082 C9ZSE5 54585303 IC50 = 38000 nM T30082 CI0ZK3 54585324 IC50 = 25500 nM T30082 C2SQ7Y 54586227 IC50 = 60 nM T30082 CNEB14 54586228 IC50 = 76 nM T30082 C97ESH 54586244 IC50 = 90 nM T30082 CUR47F 54587253 IC50 = 3 nM T30082 CY9X6B 54587254 IC50 = 70 nM T30082 CYI28B 54587266 IC50 = 16600 nM T30082 C0WMB8 54587272 IC50 = 35000 nM T30082 C8PH1A 54587274 IC50 = 2000 nM T30082 CV3F8K 54587276 IC50 = 35000 nM T30082 C75HCV 54587283 IC50 > 10000 nM T30082 C9KL7N 54587284 IC50 > 10000 nM T30082 CQ4AF0 54587306 IC50 = 26700 nM T30082 C95RDQ 54587307 IC50 = 24200 nM T30082 C2HC4E 54587308 IC50 = 25800 nM T30082 C3Y1NF 54604881 IC50 = 4300 nM T30082 C4JOA7 54753261 IC50 = 2200 nM T30082 CE1ZN5 54754513 IC50 = 9400 nM T30082 CQ1MY9 54768917 IC50 = 68.9 nM T30082 C61LVE 54768918 IC50 = 44.5 nM T30082 C6FD9U 54768919 IC50 = 16.5 nM T30082 CD19BL 54768920 IC50 = 34 nM T30082 CVQ80D 54768921 IC50 = 28.4 nM T30082 CSUP59 54768922 IC50 = 283 nM T30082 CAP3I8 54769156 IC50 = 310 nM T30082 C9O1JY 54769157 IC50 = 258 nM T30082 CQGN95 56598864 IC50 = 4500 nM T30082 C5D6ZC 56598865 IC50 = 5900 nM T30082 C26AHW 56598866 IC50 = 1700 nM T30082 CF5X9W 56600472 IC50 = 2700 nM T30082 CU2H4J 56600473 IC50 = 3100 nM T30082 CFYX02 56649564 IC50 = 45500 nM T30082 C9PQJ2 56658286 IC50 = 32200 nM T30082 C07IWL 56658287 IC50 = 31300 nM T30082 CFZ5J8 56659293 IC50 = 1800 nM T30082 CVC12H 56661785 IC50 = 15800 nM T30082 CQD4G3 56661786 IC50 = 50800 nM T30082 CV6NP7 56661787 IC50 = 11700 nM T30082 CRBY79 56661788 IC50 = 20300 nM T30082 C8H6JT 56665231 IC50 = 42500 nM T30082 CTQK07 56665232 IC50 > 100000 nM T30082 C4SEV5 56668687 IC50 = 16700 nM T30082 CY1BJ3 56668688 IC50 = 19000 nM T30082 CW9V2I 56668689 IC50 = 21600 nM T30082 CIAR59 56672159 IC50 = 13800 nM T30082 CIN62T 56672160 IC50 = 17500 nM T30082 CH7C9U 56672161 IC50 = 14600 nM T30082 CQO23H 56673143 IC50 = 6100 nM T30082 CZ5TB2 56675546 IC50 = 39200 nM T30082 CP1ZI9 56678881 IC50 = 9800 nM T30082 C4F1OQ 56678882 IC50 = 29000 nM T30082 CS48IB 56682198 IC50 = 13700 nM T30082 C9TNA0 56926078 IC50 = 17200 nM T30082 CH46AD 56926079 IC50 = 24400 nM T30082 CJ31RE 56930476 IC50 = 2.66 nM T30082 CNYF34 56930477 IC50 = 192000 nM T30082 C0J2NP 56930478 IC50 = 74100 nM T30082 CDQ32W 56933910 IC50 > 100000 nM T30082 CXNJ86 56933912 IC50 > 100000 nM T30082 CLB67G 56934051 IC50 > 100000 nM T30082 C4ZBA5 56934056 IC50 > 100000 nM T30082 C2HT1W 56935716 IC50 = 7700 nM T30082 CMA7L0 56954888 IC50 = 0.3 nM T30082 C4M1ET 56954890 IC50 = 0.775 nM T30082 C8XCI0 56954891 IC50 = 0.1 nM T30082 CHV8U3 56954986 IC50 = 2.3 nM T30082 CV3X9D 56954987 IC50 = 0.35 nM T30082 C0JCZ2 56954989 IC50 = 1.8 nM T30082 CTB71C 56954996 IC50 = 17.5 nM T30082 C4A6LW 56955097 IC50 = 0.2 nM T30082 CC7Y5O 56955099 IC50 = 8 nM T30082 C25KBX 56955100 IC50 = 1 nM T30082 C9XO0M 56955109 IC50 = 1 nM T30082 COE65B 56955111 IC50 = 2.3 nM T30082 C4U9FZ 56955198 IC50 = 0.035 nM T30082 C9I3AY 56955199 IC50 = 0.065 nM T30082 C2EY4O 56955292 IC50 = 6.5 nM T30082 C2M6DQ 56955293 IC50 = 0.09 nM T30082 C6FKT4 57339581 IC50 = 2.3 nM T30082 CL45WN 57345320 IC50 > 30000 nM T30082 CVK98Q 57383995 IC50 = 74.9 nM T30082 CHB7N4 57390352 IC50 = 11580 nM T30082 CNM3O8 57390398 IC50 = 4600 nM T30082 CD52CA 57391118 IC50 = 5600 nM T30082 CZDN40 57391125 IC50 = 89100 nM T30082 CFBU32 57391511 IC50 = 43600 nM T30082 COAM20 57392136 IC50 = 12260 nM T30082 CM31YH 57393003 IC50 = 275 nM T30082 C5D7HF 57396286 IC50 = 0.471 nM T30082 C2ZJ1Y 57396496 IC50 = 0.236 nM T30082 CJE63A 57397445 IC50 = 21100 nM T30082 C8GAU3 57398511 IC50 = 65000 nM T30082 CZ3KT7 57402629 IC50 = 18350 nM T30082 CSB12K 57405784 IC50 = 1900 nM T30082 C9F3NW 57405785 IC50 = 4200 nM T30082 C31RES 57405786 IC50 = 6100 nM T30082 C9BRL0 57405787 IC50 = 4100 nM T30082 C0RWT6 57405788 IC50 = 2500 nM T30082 CAIG86 57405951 IC50 = 3800 nM T30082 C5OWG0 57405952 IC50 = 2600 nM T30082 CK87CH 57405953 IC50 = 5100 nM T30082 C79QGF 57405954 IC50 = 5600 nM T30082 C9BKF1 57405955 IC50 = 2100 nM T30082 COU3J6 57405956 IC50 = 4700 nM T30082 C6WNC7 57406127 IC50 = 5400 nM T30082 COM8C3 57406128 IC50 = 3800 nM T30082 CQ9U4I 57406129 IC50 = 6800 nM T30082 CI65QR 57520592 IC50 = 22900 nM T30082 CRWH42 57521363 IC50 = 11.64 nM T30082 CDXQ72 58266334 IC50 = 890 nM T30082 CRZ21K 58266341 IC50 = 450 nM T30082 CV89NE 58266367 IC50 = 160 nM T30082 CL5H9F 58266371 IC50 = 187 nM T30082 C3BMF9 58266373 IC50 = 217 nM T30082 C54OAK 58266384 IC50 = 3330 nM T30082 CGX93Z 58266397 IC50 = 4100 nM T30082 CRP98K 58266398 IC50 = 2690 nM T30082 CT9U4W 58266401 IC50 = 777 nM T30082 C8RVJ3 58266453 IC50 = 708 nM T30082 CIY05G 58266579 IC50 = 323 nM T30082 CG5X8N 58266605 IC50 = 11 nM T30082 CO72RU 58266637 IC50 = 2420 nM T30082 C6YJ2E 58266718 IC50 = 266 nM T30082 CL0F3T 58266741 IC50 = 378 nM T30082 C8HT0J 58266791 IC50 = 874 nM T30082 CT42VW 58266828 IC50 = 4770 nM T30082 C6W7PQ 58266840 IC50 = 507 nM T30082 CPUM70 59740711 IC50 = 88920 nM T30082 CV2G0U 60144120 IC50 = 650 nM T30082 C4F1PE 60165327 IC50 = 3801.89 nM T30082 COIR78 60167502 IC50 = 437 nM T30082 C90BDI 60201713 IC50 = 2010 nM T30082 CO58SL 60661850 IC50 > 100000 nM T30082 C4KS0V 62707049 IC50 = 119 nM T30082 CNW04I 62707050 IC50 = 89.5 nM T30082 C1U2FD 62707051 IC50 = 139 nM T30082 C0BP3T 63753688 IC50 = 591 nM T30082 CKH2V1 63754238 IC50 = 77.5 nM T30082 CHK02P 63754964 IC50 = 6.47 nM T30082 CG14WB 63755329 IC50 = 6.11 nM T30082 CZV81L 64338500 IC50 > 100000 nM T30082 C43RLJ 65419662 IC50 = 350100 nM T30082 C60MFG 65421836 IC50 = 340200 nM T30082 CHC9K5 66561652 IC50 = 520 nM T30082 CH2E3B 66561653 IC50 = 890 nM T30082 CES43P 66561654 IC50 = 350 nM T30082 CFZ76H 66561655 IC50 = 510 nM T30082 CYRU28 66573467 IC50 = 300 nM T30082 CDVT38 66573526 IC50 = 400 nM T30082 CSA1R0 66573527 IC50 = 7830 nM T30082 CN0H5V 66573528 IC50 = 4530 nM T30082 CE52KG 66573529 IC50 = 330 nM T30082 CMXZ21 66573530 IC50 = 370 nM T30082 CC9Z1H 66573531 IC50 = 3510 nM T30082 C3W0YV 66573584 IC50 = 5740 nM T30082 C9QK4S 66573585 IC50 = 4010 nM T30082 C32IQA 66573586 IC50 = 5070 nM T30082 C0YE1R 68259803 IC50 = 2860 nM T30082 CW6ZL8 69515123 IC50 = 1030 nM T30082 C9IBN5 70681952 IC50 = 10300 nM T30082 CJ7M5L 70683121 IC50 = 1.38 nM T30082 CI03XR 70684068 IC50 = 12900 nM T30082 C09ICA 70684451 Ki = 24.7 nM T30082 CD16OS 70684889 IC50 = 240 nM T30082 CPO69B 70685195 IC50 = 0.42 nM T30082 C9HE4I 70685196 IC50 = 0.31 nM T30082 CL1EZ3 70686213 IC50 = 7700 nM T30082 CXY5N6 70686590 Ki = 1.35 nM T30082 CN8XT5 70687043 IC50 = 220 nM T30082 C4J2VL 70687142 IC50 = 9300 nM T30082 CN49BX 70687354 IC50 = 15600 nM T30082 COV1W3 70687579 IC50 = 71 nM T30082 C2B6KP 70688334 IC50 = 9900 nM T30082 C5WOI8 70689140 IC50 = 9.4 nM T30082 CZL69Q 70689406 IC50 = 316300 nM T30082 C7LMF4 70689416 IC50 = 0.89 nM T30082 CE4OI8 70689417 IC50 = 0.74 nM T30082 CV1DC5 70689418 IC50 = 1.32 nM T30082 CN8ZQ9 70690351 IC50 = 7700 nM T30082 CWT83E 70690352 IC50 = 9900 nM T30082 CU2XC0 70690775 Ki = 10.3 nM T30082 C8RPA4 70692911 Ki = 0.318 nM T30082 CC3Y2P 70692912 Ki = 13.7 nM T30082 CW8AX2 70692913 IC50 = 4.49 nM T30082 C6AHB9 70693333 IC50 = 8800 nM T30082 CA7CP6 70693341 IC50 = 120 nM T30082 C1CLT7 70694566 IC50 = 8800 nM T30082 CVG1W5 70694577 IC50 = 12600 nM T30082 C2LV8M 70694951 IC50 = 194 nM T30082 CC39LU 70695442 IC50 = 390 nM T30082 C1U2SF 70695443 IC50 = 70 nM T30082 C9XRE0 70695509 IC50 = 10800 nM T30082 CZM2Q7 70695510 IC50 = 2250 nM T30082 CZ3A8Q 70695957 IC50 = 5290 nM T30082 CY03PS 70696614 IC50 = 9400 nM T30082 CF9EO8 70697005 Ki = 16.8 nM T30082 CWO7H5 70697453 IC50 = 3100 nM T30082 CZT65E 71081197 IC50 = 63000 nM T30082 CCG8L7 71088584 IC50 > 20000 nM T30082 CN93VA 71330901 IC50 = 6300 nM T30082 C7AJN9 71449137 IC50 = 0.32 nM T30082 CRC86Q 71449660 Ki = 45.81 nM T30082 CVF86W 71449711 IC50 = 102000 nM T30082 CE9MV7 71451470 Ki = 1437 nM T30082 C24OJQ 71451471 Ki = 123.73 nM T30082 CVKC68 71451473 Ki = 81 nM T30082 C7NS9H 71451521 IC50 = 53000 nM T30082 CDES68 71451522 IC50 = 78000 nM T30082 CJG67A 71452919 IC50 = 4.04 nM T30082 CAMW73 71453296 Ki > 10000 nM T30082 C5CK7V 71453297 Ki = 6.47 nM T30082 CYVB31 71453347 IC50 = 215000 nM T30082 CTJ6W4 71453348 IC50 = 340 nM T30082 C28XSH 71454519 IC50 = 0.29 nM T30082 C4JDI7 71455058 IC50 = 240 nM T30082 CAJ7O6 71456744 Ki = 3520 nM T30082 C0RNU7 71456800 Ki > 10000 nM T30082 CL02JI 71456801 Ki = 53 nM T30082 CC7F6N 71456803 Ki = 44.66 nM T30082 C2B8LY 71456805 Ki = 9.4 nM T30082 C1D6KG 71456857 IC50 = 101000 nM T30082 CP4K8E 71456859 IC50 = 39000 nM T30082 C16BOY 71458659 Ki > 10000 nM T30082 CFN68Z 71458660 Ki > 10000 nM T30082 CH7L4U 71458714 IC50 = 67700 nM T30082 C35XHD 71458715 IC50 = 37100 nM T30082 C36LDS 71460126 IC50 = 5.18 nM T30082 CLF31N 71460483 Ki > 10000 nM T30082 CXHM16 71460484 Ki = 197.78 nM T30082 CXIQ97 71461841 IC50 = 3.52 nM T30082 C2JBI7 71462190 Ki = 47 nM T30082 CBM3S6 71462240 IC50 = 100000 nM T30082 C6S5WO 71462637 IC50 = 3000 nM T30082 C63NIZ 71481105 Ki = 55180 nM T30082 C8OL3N 71482804 IC50 = 4602.57 nM T30082 CGC2I3 71492939 Ki = 3178000 nM T30082 CV17CS 71492940 Ki = 2430000 nM T30082 C64XWL 71492941 Ki = 266000 nM T30082 CVQ4I2 71492943 Ki = 1492 nM T30082 CRC0U4 71492944 Ki = 588.1 nM T30082 CZAV42 71493110 Ki = 31220 nM T30082 C6E1LN 71493111 Ki = 198500 nM T30082 CE8HA0 71493283 Ki = 732500 nM T30082 CKA54I 71493285 Ki = 94963000 nM T30082 C43UGA 71533432 Ki = 19500 nM T30082 CO6IV1 71533433 Ki = 50800 nM T30082 CRA7K6 71540497 IC50 = 62800 nM T30082 C21QXB 71584433 IC50 = 17390 nM T30082 CFNK45 71584434 IC50 = 8720 nM T30082 C5AP4Q 71584435 IC50 = 11810 nM T30082 CON9H3 71584436 IC50 = 9760 nM T30082 CLN29O 71587645 IC50 = 110 nM T30082 CN1X5W 71602710 IC50 = 1760 nM T30082 CLJ71T 71614508 IC50 = 13840 nM T30082 CDM3U5 71614509 IC50 = 15720 nM T30082 C62PLB 71614697 IC50 = 11200 nM T30082 CC41TG 71614698 IC50 = 14520 nM T30082 C7X0TU 71614699 IC50 = 5080 nM T30082 CWVY13 71614700 IC50 = 29510 nM T30082 C3ECM4 71614898 IC50 = 4280 nM T30082 CT4Q6N 71614899 IC50 = 3330 nM T30082 C6U3GL 71614900 IC50 = 7600 nM T30082 CXF97V 71614901 IC50 = 3360 nM T30082 C35WPQ 71615100 IC50 = 22320 nM T30082 CC75NE 71615101 IC50 = 5810 nM T30082 C6DB9K 71699482 IC50 = 92 nM T30082 C3VO0M 71716370 IC50 = 26600 nM T30082 C7A1KW 71716371 IC50 = 24580 nM T30082 C09HUL 71716383 IC50 = 20630 nM T30082 CFWE09 71716757 IC50 = 43 nM T30082 CH72KQ 71716973 IC50 = 12470 nM T30082 CD2F8T 71716974 IC50 = 15860 nM T30082 C73XHB 71716985 IC50 = 34370 nM T30082 C85WCB 71716986 IC50 = 4110 nM T30082 CSCF90 71716987 IC50 = 3360 nM T30082 CP82JA 71717595 IC50 = 7920 nM T30082 C58SQT 71718212 IC50 = 19590 nM T30082 CK2Q5O 71718812 IC50 = 16320 nM T30082 CRME79 71718813 IC50 = 6760 nM T30082 CMA97I 71718814 IC50 = 17490 nM T30082 CQM0H7 71718831 IC50 = 11920 nM T30082 CIT85H 71719411 IC50 = 6960 nM T30082 C6WNO7 71719412 IC50 = 11410 nM T30082 C9V4DF 71719421 IC50 = 20070 nM T30082 CVC3A2 71720009 IC50 = 23670 nM T30082 CON03A 71720010 IC50 = 19650 nM T30082 CQX83T 71720016 IC50 = 5990 nM T30082 CY0FN4 71720017 IC50 = 19840 nM T30082 CM9DZ3 71720635 IC50 = 13640 nM T30082 CQD35G 71720636 IC50 = 27450 nM T30082 C2VE3P 71720637 IC50 = 15750 nM T30082 CFMB35 71723450 IC50 > 100000 nM T30082 CV16HS 71723451 IC50 > 100000 nM T30082 C7U5ER 71723452 IC50 > 100000 nM T30082 CF2VL4 71723589 IC50 = 59680 nM T30082 COT21H 71723590 IC50 > 100000 nM T30082 CA6ZR8 71732757 IC50 = 5395.11 nM T30082 C8I3MR 71740897 IC50 = 190 nM T30082 CL5Y3O 71740898 IC50 = 690 nM T30082 CVPF08 71769270 IC50 = 10680 nM T30082 CIC3T9 71769271 IC50 > 100000 nM T30082 C0B7VI 71769272 IC50 = 23420 nM T30082 C5ADC9 71769273 IC50 = 2130 nM T30082 C03DUA 71769382 IC50 > 100000 nM T30082 C8N0VS 71769383 IC50 = 12340 nM T30082 CT9BD7 71769384 IC50 = 50980 nM T30082 CL2I3N 71769385 IC50 = 400 nM T30082 C3YQW9 71769386 IC50 = 390 nM T30082 CE7J6B 71769387 IC50 = 12920 nM T30082 C06MNJ 71769388 IC50 = 8020 nM T30082 CXP9U3 71769495 IC50 = 3680 nM T30082 CHYB71 71769496 IC50 = 1400 nM T30082 C56ZQT 71769497 IC50 = 130 nM T30082 CV2EY6 71769498 IC50 = 9730 nM T30082 CAV41T 71816334 IC50 = 11940 nM T30082 CYE81W 72192858 IC50 = 20900 nM T30082 CTN81V 72193164 IC50 = 12100 nM T30082 C4R9EZ 72374595 IC50 = 13 nM T30082 CK38PO 72374596 IC50 = 4400 nM T30082 C0FN4W 72374597 IC50 = 9770 nM T30082 CC5E6T 72374847 IC50 = 810 nM T30082 C73ATU 72374849 IC50 = 100 nM T30082 CE2W4A 72374851 IC50 = 70 nM T30082 C0VM3N 72374853 IC50 = 120 nM T30082 C8J5VN 72374855 IC50 = 180 nM T30082 C4IPA8 72374968 IC50 = 5200 nM T30082 CHG4A5 72374970 IC50 = 460 nM T30082 CMG0R4 72374972 IC50 = 190 nM T30082 CY9PG6 72374974 IC50 = 49 nM T30082 CXVJ78 72375088 IC50 = 130 nM T30082 CK8N5F 72375090 IC50 = 70 nM T30082 CN9M6L 72375092 IC50 = 190 nM T30082 CIUG39 72375094 IC50 = 98000 nM T30082 CF14AL 72375096 IC50 = 3600 nM T30082 CCG9N8 72375206 IC50 = 22000 nM T30082 C2ED8X 72375208 IC50 = 3600 nM T30082 CBHY20 72375210 IC50 = 760 nM T30082 CP0G4A 72375212 IC50 = 720 nM T30082 CK14WV 72375214 IC50 = 1700 nM T30082 C70BZS 72375315 IC50 = 530 nM T30082 C0ZW8S 72375317 IC50 = 470 nM T30082 C9LNA8 72376170 IC50 = 3860 nM T30082 CULW84 72376171 IC50 = 31 nM T30082 CY19TH 72376172 IC50 = 54 nM T30082 C45BXP 72543919 IC50 = 600 nM T30082 C78ZPH 72544154 IC50 = 9540 nM T30082 CKAG40 72544155 IC50 = 600 nM T30082 CPH96F 72544156 IC50 = 10300 nM T30082 CE49KY 72544381 IC50 > 20000 nM T30082 CTW28Y 72544382 IC50 = 107000 nM T30082 C6TQ7M 72545286 IC50 = 27800 nM T30082 CBL6J5 72545287 IC50 = 2890 nM T30082 CH41BM 72696518 IC50 = 98 nM T30082 CY9NX6 72696519 IC50 = 156.8 nM T30082 C4LCA1 72696649 IC50 = 121.6 nM T30082 CS5J3B 72696781 IC50 = 105.3 nM T30082 C3H2IR 72714446 IC50 = 23000 nM T30082 CEIW98 72724703 IC50 = 15.13 nM T30082 CKY67A 72724835 IC50 = 800 nM T30082 C59UPS 72724837 IC50 = 140 nM T30082 CA16UV 72724839 IC50 = 40 nM T30082 CTB2A1 72724841 IC50 = 20 nM T30082 C02IHQ 72724843 IC50 = 30 nM T30082 CGJ2T1 72724905 IC50 = 540 nM T30082 C5Z4BW 72724907 IC50 = 270 nM T30082 CJA54D 72724909 IC50 = 120 nM T30082 C3OUZ2 72724911 IC50 = 5 nM T30082 CY2M3K 72724913 IC50 = 17 nM T30082 CPWA14 72724915 IC50 = 4.7 nM T30082 C1LH5Z 72725438 Ki = 0.78 nM T30082 C6CJT1 72725439 Ki = 0.23 nM T30082 C3K0SD 72725440 Ki = 1.92 nM T30082 CS1TQ7 72725488 Ki = 5.02 nM T30082 C9ZB1M 72725489 Ki = 1.48 nM T30082 C7P3NJ 72725625 IC50 = 19.52 nM T30082 CL1ZH8 72736377 IC50 = 231 nM T30082 C0P7RN 72736548 IC50 = 103 nM T30082 CEK38F 72736549 IC50 = 163 nM T30082 CNK69L 72736878 IC50 = 97 nM T30082 C9IB7C 73345791 IC50 = 1780 nM T30082 C86QTX 73345830 IC50 = 1780 nM T30082 CVF16T 73345831 IC50 = 1780 nM T30082 C53XHE 73346133 IC50 = 310 nM T30082 C0WB1S 73347274 IC50 = 1780 nM T30082 C81JUL 73348052 IC50 = 36000 nM T30082 CG4Q6E 73348054 IC50 = 21000 nM T30082 CO26TZ 73349587 IC50 = 70000 nM T30082 CEM3S7 73349589 IC50 = 16000 nM T30082 C9RWV8 73352248 IC50 = 9430 nM T30082 COKX05 73352249 IC50 = 7300 nM T30082 CQJC68 73353352 IC50 = 1780 nM T30082 C0H4PZ 73353389 IC50 = 1780 nM T30082 CMTD19 73354116 IC50 = 7500 nM T30082 C8Z6CW 73354118 IC50 = 51000 nM T30082 C6I8BF 73354120 IC50 = 43000 nM T30082 C9HU8K 73354122 IC50 = 14000 nM T30082 CJR13W 73354173 IC50 = 62 nM T30082 CCM7N1 73354902 IC50 = 1780 nM T30082 C5T7SG 73354903 IC50 = 1780 nM T30082 CHZ9S6 73355637 IC50 = 54000 nM T30082 CIG0U4 73356417 IC50 = 344 nM T30082 CR6G8D 73356461 IC50 = 1780 nM T30082 C45GXL 73356781 IC50 = 5350 nM T30082 CGD8R4 73671789 IC50 = 350 nM T30082 CE8T5U 76285505 IC50 = 10520 nM T30082 CEZ0N5 76285506 IC50 = 1440 nM T30082 CFQ92C 76307955 IC50 = 3890.45 nM T30082 CV7SH8 76307956 IC50 = 69183.1 nM T30082 CFVN49 76307957 IC50 = 7079.46 nM T30082 C8TPQ6 76307958 IC50 = 602.56 nM T30082 C1V3TM 76307959 IC50 = 27542.29 nM T30082 C2UCN8 76307984 IC50 = 1698.24 nM T30082 CZ06NV 76307985 IC50 = 8511.38 nM T30082 CF2H4Q 76307986 IC50 = 23988.33 nM T30082 C0SL7X 76307987 IC50 = 1819.7 nM T30082 C7P2ZK 76310594 IC50 = 5190 nM T30082 CA20OP 76310595 IC50 = 4100 nM T30082 CI2J8H 76310596 IC50 = 8400 nM T30082 CV13PU 76310709 IC50 = 6700 nM T30082 CDM6R7 76310865 IC50 > 25000 nM T30082 C5PLC4 76310867 IC50 = 13000 nM T30082 CA4TK7 76311545 IC50 = 1905.46 nM T30082 C1WYH4 76311546 IC50 = 19054.61 nM T30082 C36ERB 76311573 IC50 = 26915.35 nM T30082 CH9C4D 76311574 IC50 = 20892.96 nM T30082 C86SDL 76311575 IC50 = 3467.37 nM T30082 CU4Y5V 76311843 IC50 = 8240 nM T30082 CNH0V3 76314228 IC50 = 4310 nM T30082 CH2IJ4 76314229 IC50 = 450 nM T30082 C7R3UV 76314230 IC50 > 15000 nM T30082 CKF2X0 76314231 IC50 = 7800 nM T30082 CZDB68 76314491 IC50 = 1060 nM T30082 CEMK74 76314492 IC50 > 25000 nM T30082 C0P4EI 76314828 IC50 = 330 nM T30082 C39CVT 76314829 IC50 = 2430 nM T30082 CE8LX0 76315115 IC50 = 2137.96 nM T30082 C9TXY2 76315116 IC50 = 93325.43 nM T30082 C3V8LC 76315117 IC50 = 537.03 nM T30082 CL48SJ 76315118 IC50 = 6606.93 nM T30082 C8YB3A 76315135 IC50 = 32359.37 nM T30082 C4PYG8 76315136 IC50 = 4570.88 nM T30082 CN03PG 76315137 IC50 = 1548.82 nM T30082 CB3SK9 76315267 IC50 = 0.82 nM T30082 C56PFG 76315394 IC50 = 10130 nM T30082 C74HJI 76317800 IC50 > 15000 nM T30082 C9JV1O 76317801 IC50 = 3410 nM T30082 CYC3S2 76317802 IC50 = 6180 nM T30082 C62TKJ 76317803 IC50 = 6140 nM T30082 CGI2O5 76317912 IC50 = 2900 nM T30082 C1I2UO 76317913 IC50 > 10000 nM T30082 CE5M1O 76317914 IC50 > 10000 nM T30082 CC1PL3 76318071 IC50 = 556 nM T30082 C8REX0 76318435 IC50 = 2440 nM T30082 CG0UV3 76318770 IC50 = 1862.09 nM T30082 CJ3MA9 76318771 IC50 = 51286.14 nM T30082 CX5I1F 76318772 IC50 = 79.43 nM T30082 C4RMS6 76318773 IC50 = 323.59 nM T30082 C8VA5B 76318774 IC50 = 229.09 nM T30082 CDKN48 76318775 IC50 = 16982.44 nM T30082 CNC7P9 76319071 IC50 = 7030 nM T30082 CV4W1T 76319072 IC50 = 19090 nM T30082 C9XB6I 76319073 IC50 = 7690 nM T30082 CY6X4K 76321510 IC50 = 10930 nM T30082 CW0UI6 76321511 IC50 = 4730 nM T30082 C9FHG6 76321512 IC50 = 5120 nM T30082 C4M8ZY 76321622 IC50 = 7100 nM T30082 CSXH87 76321623 IC50 > 10000 nM T30082 C35UQW 76321779 IC50 > 25000 nM T30082 CF28AB 76321780 IC50 = 4150 nM T30082 C6O5XW 76321781 IC50 > 25000 nM T30082 CF9BX2 76322101 IC50 = 930 nM T30082 CU24PD 76322416 IC50 = 21379.62 nM T30082 C3ZIQ9 76322417 IC50 = 158.49 nM T30082 CL5RQ7 76322452 IC50 = 14454.4 nM T30082 C7HD5Z 76322453 IC50 = 7762.47 nM T30082 C1YXL9 76322454 IC50 = 1949.84 nM T30082 CUYZ32 76322728 IC50 = 6580 nM T30082 C7CG1Q 76322729 IC50 = 9370 nM T30082 C4ULY3 76325115 IC50 = 4420 nM T30082 CYR12G 76325116 IC50 = 7670 nM T30082 CA47NE 76325117 IC50 = 6140 nM T30082 C1W8HB 76325234 IC50 > 10000 nM T30082 CO05NW 76325235 IC50 > 25000 nM T30082 C8DSR5 76325563 IC50 = 3880 nM T30082 CK2EG4 76325714 IC50 = 870 nM T30082 CZ9P6V 76325715 IC50 = 2990 nM T30082 C9CRD3 76326035 IC50 = 3890.45 nM T30082 CG3NZ7 76326036 IC50 = 602.56 nM T30082 CSB53W 76326037 IC50 = 91.2 nM T30082 CT0Z1Y 76326038 IC50 = 61.66 nM T30082 C2K7CE 76326039 IC50 = 12882.5 nM T30082 CU3NO7 76326040 IC50 = 21877.62 nM T30082 CEL04N 76326288 IC50 = 8050 nM T30082 CN82AX 76328677 IC50 = 13940 nM T30082 CAOR72 76328678 Ki = 2010 nM T30082 CK8ZH0 76328679 IC50 = 4930 nM T30082 CS42NU 76328680 IC50 = 3970 nM T30082 CR5VT1 76328681 IC50 = 7490 nM T30082 C5AV9G 76328789 IC50 > 10000 nM T30082 C4QH5I 76328790 IC50 > 10000 nM T30082 C30AMV 76328791 IC50 = 91000 nM T30082 CB1KJ6 76328792 IC50 > 10000 nM T30082 CEKP26 76328944 IC50 = 15800 nM T30082 CL94XO 76328945 IC50 > 25000 nM T30082 CUE86C 76329116 IC50 = 350 nM T30082 CD52FV 76329288 IC50 = 1130 nM T30082 C92XLS 76329623 IC50 = 48977.88 nM T30082 CUO23D 76329624 IC50 = 109.65 nM T30082 C3RD8U 76329625 IC50 = 14125.38 nM T30082 CC9AL5 76329626 IC50 = 870.96 nM T30082 CFJ2H7 76329644 IC50 = 7079.46 nM T30082 CP3I4S 76329645 IC50 = 24547.09 nM T30082 C6SY7C 76329646 IC50 = 12882.5 nM T30082 CRT50O 76329906 IC50 = 3250 nM T30082 CQH6C3 76329907 IC50 = 23140 nM T30082 C12RPG 76332357 IC50 = 5150 nM T30082 CZL0S8 76332358 IC50 = 10850 nM T30082 CC2L9I 76332359 IC50 = 2470 nM T30082 C1EPW9 76332360 IC50 = 6880 nM T30082 CS61PT 76332365 IC50 = 7590 nM T30082 CJ8O4M 76332773 IC50 = 5800 nM T30082 CCUL46 76332937 IC50 = 1320 nM T30082 C2ZDE5 76332939 IC50 = 880 nM T30082 C39KJU 76332940 IC50 = 9180 nM T30082 CIP03O 76333286 IC50 = 17782.79 nM T30082 COTJ98 76333287 IC50 = 12022.64 nM T30082 CVAC53 76333288 IC50 = 40738.03 nM T30082 CVLM78 76333289 IC50 = 52.48 nM T30082 C1GTV7 76333290 IC50 = 302 nM T30082 C1TMA2 76333291 IC50 = 218.78 nM T30082 CKC1H8 76333292 IC50 = 16982.44 nM T30082 CNG40D 76333293 IC50 = 3019.95 nM T30082 CY4UJ2 76333319 IC50 = 33113.11 nM T30082 C1LZA6 76333438 IC50 = 0.32 nM T30082 C4EKP8 76333548 IC50 = 7100 nM T30082 CM2T5R 76333549 IC50 = 10360 nM T30082 C7XHK6 76333550 IC50 = 17560 nM T30082 CJ3HD4 76335987 IC50 = 8740 nM T30082 C5IAN4 76335988 IC50 = 5340 nM T30082 C2EU0T 76335993 IC50 = 2630 nM T30082 CFY2O3 76335994 IC50 = 9430 nM T30082 CTG51J 76336093 IC50 > 10000 nM T30082 CO8FB2 76336222 Ki = 785 nM T30082 C1BN8V 76336223 IC50 = 942 nM T30082 CW8Y5E 76336226 IC50 = 22800 nM T30082 C48RZI 76336227 IC50 = 65 nM T30082 CEO54B 76336549 IC50 = 1840 nM T30082 C57UTS 77108165 IC50 = 800 nM T30082 C0JCK7 77461631 IC50 > 10000 nM T30082 CH5YI4 77844667 IC50 = 78300 nM T30082 CDJ5S9 78319301 IC50 = 2530000 nM T30082 C4BM2W 78319305 IC50 = 1700000 nM T30082 C45KVG 78319307 IC50 = 2100000 nM T30082 C7GX5I 78350462 IC50 = 0.72 nM T30082 CA3YL2 78426937 IC50 = 2800 nM T30082 CR0H5Q 78427074 IC50 = 6000 nM T30082 C2ZOJ4 78427075 IC50 = 1300 nM T30082 CJCL87 78427076 IC50 = 2100 nM T30082 CH3NJ9 78427077 IC50 = 2700 nM T30082 CR84AG 78427078 IC50 = 4300 nM T30082 CV9DO7 78427079 IC50 = 4900 nM T30082 C4US9B 78427204 IC50 = 900 nM T30082 CS0N1V 78427205 IC50 = 1000 nM T30082 CG46NS 78427206 IC50 = 1700 nM T30082 C3WL0E 78427207 IC50 = 6400 nM T30082 CK5X0H 78427208 IC50 = 900 nM T30082 CN6L8C 78427209 IC50 = 4100 nM T30082 CCE8Q9 78427338 IC50 = 1100 nM T30082 C14JGF 80099174 IC50 = 2.27 nM T30082 C0CL4Y 80772460 IC50 = 8700 nM T30082 CI5GO1 83453608 IC50 = 2300 nM T30082 C5MC7H 85470203 IC50 > 10000 nM T30082 CHXN26 85852196 Ki = 11800 nM T30082 C7IK2X 86276151 Ki = 232600 nM T30082 C23XGV 86276159 Ki = 180100 nM T30082 CIB29V 86279207 IC50 = 230 nM T30082 CEW6N9 86279208 IC50 = 980 nM T30082 C7IWL1 86287984 IC50 = 3660 nM T30082 CE6S1P 86287985 IC50 = 2320 nM T30082 CB3ZI5 86294786 IC50 = 2200 nM T30082 CXC80P 86581945 IC50 = 59 nM T30082 CZ75NQ 86582973 Ki = 16 nM T30082 CR85FW 87056148 IC50 = 63.2 nM T30082 C8CF5A 88749792 IC50 > 100000 nM T30082 CD6Q5Y 89400859 Ki = 6219 nM T30082 CRN2F3 89969848 Ki = 137400 nM T30082 CP3X6I 89969871 Ki = 344800 nM T30082 CI27SD 89969881 Ki = 285600 nM T30082 CTYX60 89969946 Ki = 2517000 nM T30082 CSA16V 89969958 Ki = 595100 nM T30082 CMA40S 89969964 Ki = 1930000 nM T30082 CX8GS4 89969971 Ki = 144000 nM T30082 C1XQV0 89969999 Ki = 199100 nM T30082 CG57IR 89972500 Ki = 3077 nM T30082 CRZ0W3 90356636 IC50 = 8500 nM T30082 CI3ZW5 90356648 IC50 = 18000 nM T30082 C85UDM 90356741 IC50 = 27400 nM T30082 C2Z5FB 90356750 IC50 = 8200 nM T30082 CYB89Q 90356760 IC50 = 6700 nM T30082 CW8N4S 90356765 IC50 = 29300 nM T30082 C3NKB2 90356879 IC50 = 20900 nM T30082 CO1RJ4 90356882 IC50 = 13700 nM T30082 C9UI0O 90356903 IC50 = 20000 nM T30082 CO2HX6 90356923 IC50 = 8300 nM T30082 C52SQL 90356955 IC50 = 18500 nM T30082 C5YD7M 90356964 IC50 = 18400 nM T30082 C31XOK 90357088 IC50 = 11400 nM T30082 C0P3IL 90357101 IC50 = 7300 nM T30082 CR54TH 90357102 IC50 = 10900 nM T30082 CBJ4I2 90357105 IC50 = 21300 nM T30082 CDXO02 90357107 IC50 = 15100 nM T30082 CY9T0A 90357109 IC50 = 14200 nM T30082 CWKM49 90357121 IC50 = 2800 nM T30082 CZ7CG4 90357147 IC50 = 8700 nM T30082 C1FKL7 90357154 IC50 = 8100 nM T30082 C1LO9P 90357159 IC50 = 9200 nM T30082 CYDQ90 90357180 IC50 = 37200 nM T30082 C3I9SK 90357196 IC50 = 6200 nM T30082 CSY64P 90357367 IC50 = 18900 nM T30082 CTVJ69 90645106 IC50 = 12430 nM T30082 CYW8G5 90645107 IC50 = 41220 nM T30082 C1R6LU 90645108 IC50 = 920 nM T30082 C5U8JA 90645109 IC50 = 42 nM T30082 C8CKM6 90645110 IC50 = 27540 nM T30082 CYN86M 90645111 IC50 = 55340 nM T30082 C3EAW0 90645112 IC50 = 76640 nM T30082 C4XF1V 90645113 IC50 > 100000 nM T30082 C30WLJ 90645114 IC50 > 100000 nM T30082 CG6YO8 90645115 IC50 = 76930 nM T30082 CJZ4X5 90645116 IC50 = 45290 nM T30082 CO20MQ 90645117 IC50 = 1540 nM T30082 C8QHF2 90645118 IC50 = 880 nM T30082 CVPN52 90645119 IC50 = 57 nM T30082 CXHK56 90645120 IC50 > 100000 nM T30082 CF4EB2 90645121 IC50 > 100000 nM T30082 CB2E7N 90645122 IC50 > 100000 nM T30082 CR2VS4 90645123 IC50 > 100000 nM T30082 C1ZYO3 90645124 IC50 = 79310 nM T30082 C2CI1S 90645125 IC50 = 39440 nM T30082 C40YGU 90645126 IC50 > 100000 nM T30082 C4R7BX 90645127 IC50 > 100000 nM T30082 CMN7Z9 90645128 IC50 = 9520 nM T30082 C62RBA 90645129 IC50 = 2780 nM T30082 CXU48E 90645130 IC50 > 100000 nM T30082 CYG4D2 90645131 IC50 = 66430 nM T30082 CPM6V1 90645132 IC50 > 100000 nM T30082 CP1OU8 90645133 IC50 > 100000 nM T30082 CAB7V8 90654202 IC50 = 1096.67 nM T30082 CJ6Z2M 90654884 IC50 = 130000 nM T30082 C79FOK 90654891 IC50 = 150 nM T30082 C5X2IV 90654980 IC50 = 2.15 nM T30082 CWF6X2 90654981 IC50 = 5.04 nM T30082 CMC46P 90655184 IC50 = 1.07 nM T30082 C12GDL 90655186 IC50 = 1.52 nM T30082 C36VCM 90655188 IC50 = 3.18 nM T30082 CL7PI9 90655190 IC50 = 4.36 nM T30082 CZ18NX 90655191 IC50 = 3.6 nM T30082 CH7C4F 90655192 IC50 = 2930 nM T30082 CMJ31X 90655193 IC50 = 2.39 nM T30082 C3IZ2O 90655195 IC50 = 7.61 nM T30082 CG69TU 90655196 IC50 = 17.4 nM T30082 C6WH0F 90655198 IC50 = 18.2 nM T30082 CZ14AD 90655424 IC50 > 100000 nM T30082 CEM9U7 90655425 IC50 = 17100 nM T30082 C9MLI3 90655426 IC50 > 100000 nM T30082 CP8S6V 90655427 IC50 = 71500 nM T30082 C6BJ8G 90655428 IC50 > 100000 nM T30082 CK7UE4 90655429 IC50 = 9100 nM T30082 C6KXL4 90655683 Ki = 158800 nM T30082 C0T4VJ 90655684 Ki = 1608000 nM T30082 CAT3Z9 90655685 Ki = 298300 nM T30082 CN8GU5 90655686 Ki = 550600 nM T30082 C21MQU 90656253 IC50 = 1430000 nM T30082 CLUT69 90656255 IC50 = 930000 nM T30082 C1YL8H 90656257 IC50 = 1670000 nM T30082 C4CFZ3 90656259 IC50 = 1070000 nM T30082 CM47DE 90656260 IC50 = 1060000 nM T30082 C82OEJ 90656261 IC50 = 1790000 nM T30082 CT2N6S 90656307 IC50 = 9590 nM T30082 CTXS90 90656308 IC50 = 35480 nM T30082 CHJ71K 90656309 IC50 = 39630 nM T30082 C1FSU2 90656310 IC50 = 16330 nM T30082 CMAJ10 90656311 IC50 = 5590 nM T30082 CY0KN8 90656312 IC50 = 9330 nM T30082 CF9A7K 90656313 IC50 = 4990 nM T30082 C2I0ZP 90656314 IC50 = 7130 nM T30082 CKXS95 90656315 IC50 = 3460 nM T30082 CP4D2I 90656316 IC50 = 3850 nM T30082 CDV62L 90656317 IC50 = 4500 nM T30082 C2E0NT 90656318 IC50 = 2140 nM T30082 CS4ZQ0 90656319 IC50 = 2980 nM T30082 C6JS8W 90664279 IC50 = 140 nM T30082 CY86BC 90664299 IC50 = 18.3 nM T30082 C7NGZ1 90664300 IC50 = 11.1 nM T30082 C1KOL2 90664301 IC50 = 14 nM T30082 C30SQY 90664402 Ki = 1.91 nM T30082 CKU86A 90664403 IC50 = 24.9 nM T30082 CM4NF3 90664404 IC50 = 50 nM T30082 CKL69C 90664470 IC50 = 1.89 nM T30082 CL65ZG 90664552 IC50 = 16.6 nM T30082 C0GN8Y 90664609 IC50 = 3.53 nM T30082 C05QSY 90664655 Ki = 207700 nM T30082 CPE7N6 90664658 IC50 = 2.6 nM T30082 CYGT83 90664665 IC50 = 14.4 nM T30082 CO82LG 90664779 IC50 = 0.67 nM T30082 C90OVC 90664784 IC50 = 19.2 nM T30082 C4EA8P 90664797 IC50 = 1 nM T30082 C7H6ZG 90664851 IC50 = 4.19 nM T30082 C3AON4 90664852 IC50 = 4.02 nM T30082 CI0NQ2 90664853 IC50 = 2.04 nM T30082 CLQ1F4 90664854 IC50 = 11.5 nM T30082 CFK51Z 90664907 IC50 = 0.27 nM T30082 CI1T4S 90664976 IC50 = 1.33 nM T30082 CXB25V 90664977 IC50 = 3.26 nM T30082 C1DN7L 90664978 IC50 = 9.09 nM T30082 CFPS72 90665034 Ki = 316400 nM T30082 CW36ZP 90665154 IC50 = 1.06 nM T30082 C80QZK 90665217 IC50 = 6.84 nM T30082 CAS3P4 90667148 IC50 = 41370 nM T30082 C9EDT4 90667149 IC50 = 69470 nM T30082 C1HJB5 90667151 IC50 = 15010 nM T30082 CB70OR 90667344 IC50 = 150000 nM T30082 C17ZXD 90667346 IC50 = 30000 nM T30082 C2JT9Z 90667348 IC50 = 88000 nM T30082 C8SUR1 90667350 IC50 = 2200 nM T30082 CTDR94 90667352 IC50 = 5000 nM T30082 CYIJ47 90667354 IC50 = 80000 nM T30082 C6J7ZA 90667356 IC50 = 34000 nM T30082 CTWS98 90667358 IC50 = 9000 nM T30082 C1PY0T 90676323 IC50 = 6400 nM T30082 CG9JP4 91689645 IC50 = 7500 nM T30082 C7C9RB 91689712 IC50 = 4600 nM T30082 C8NC7S 91689713 IC50 = 6400 nM T30082 CAM0G8 91864546 Ki = 0.72 nM T30082 CUPK70 91885433 IC50 = 300 nM T30082 C48VLU 92204752 IC50 = 35 nM T30082 C5RF6O 101077957 IC50 = 910 nM T30082 CV2B4X 101450543 IC50 = 2500 nM T30082 CG3E2C 101521169 IC50 = 6516.28 nM T30082 CF02IH 101521171 IC50 = 6776.42 nM T30082 CH8FU7 101521172 IC50 = 5834.45 nM T30082 C4HLR3 101528287 IC50 > 30000 nM T30082 CO6NX1 101562527 IC50 = 2150000 nM T30082 CD28FK 101562528 IC50 = 2249.05 nM T30082 C7T4UV 101562529 IC50 = 5180000 nM T30082 C8RPO5 101562530 IC50 = 389.94 nM T30082 C5FI8L 101562531 IC50 = 380.19 nM T30082 CVD19H 101803137 IC50 = 709.58 nM T30082 C5V2JH 101886788 IC50 = 1.93 nM T30082 CLO03N 101886789 IC50 = 24.7 nM T30082 CF6EI0 101886790 IC50 = 14.3 nM T30082 C52VTG 101886792 IC50 = 53.7 nM T30082 CV3A0F 101886793 IC50 = 2530 nM T30082 CI2U0Y 101886794 IC50 = 5.4 nM T30082 C56IGC 101886796 IC50 = 9.24 nM T30082 C6GL0Y 101893725 IC50 = 53000 nM T30082 C8HE3Q 101893726 IC50 = 68000 nM T30082 C6W2JF 101898808 Ki = 16.7 nM T30082 CJ47GT 101902496 IC50 = 142 nM T30082 C81WRJ 101910778 IC50 = 2800 nM T30082 CMN08X 102157796 IC50 = 75350 nM T30082 CDBZ20 102189779 IC50 = 3213 nM T30082 C1PAK7 102257397 IC50 = 4850 nM T30082 C71RIU 102257398 IC50 = 1020 nM T30082 C4XMG6 102257401 IC50 = 1250 nM T30082 C4LJ9O 102369422 IC50 = 26.3 nM T30082 CY93VO 102369423 Ki = 4.1 nM T30082 CL96MC 102532094 IC50 > 100 ug.mL-1 T30082 C58TCX 107886865 IC50 = 8.37 nM T30082 CSF32B 110298324 IC50 = 4.11 nM T30082 C74UZL 112684088 IC50 = 0.02685 nM T30082 CK52CI 112686058 Ki = 0.0049 nM T30082 CP5B7N 112687648 Ki = 0.0063 nM T30082 CT9H1Y 118557791 IC50 = 286 nM T30082 C5EH7X 118557800 IC50 = 262 nM T30082 CKOV73 118557808 IC50 = 0.36 nM T30082 CF83VS 118557818 IC50 = 568 nM T30082 CXI80V 118557824 IC50 = 18 nM T30082 C9VJK3 118557841 IC50 = 71 nM T30082 CLTV82 118557854 IC50 > 10000 nM T30082 C6NM8Z 118557858 IC50 = 428 nM T30082 C8UYK3 118557871 IC50 > 10000 nM T30082 CO09ZT 118557882 IC50 > 1000 nM T30082 CGH4F5 118557887 IC50 = 307.5 nM T30082 C8ELF0 118557908 IC50 = 29.5 nM T30082 C5P1IR 118557917 IC50 > 1000 nM T30082 CNH40Y 118557924 IC50 = 110.5 nM T30082 C0F4UC 118557927 IC50 = 43 nM T30082 C6I7SY 118557943 IC50 > 10000 nM T30082 C84WYR 118557950 IC50 = 653 nM T30082 CW59QD 118557956 IC50 > 1000 nM T30082 CZ7OM6 118557961 IC50 > 1000 nM T30082 CGI52P 118557966 IC50 > 1000 nM T30082 CD5LP8 118557967 IC50 = 10 nM T30082 C35WAU 118557974 IC50 > 10000 nM T30082 CME6H0 118557975 IC50 = 8.8 nM T30082 C8CW5V 118557990 IC50 = 30 nM T30082 CC28UL 118558001 IC50 > 10000 nM T30082 CGX48A 118558018 IC50 = 55.5 nM T30082 CU8O9N 118558025 IC50 = 3.27 nM T30082 CJDU45 118558040 IC50 = 27.7 nM T30082 CF29QK 118558043 IC50 = 60 nM T30082 C9JL5C 118558055 IC50 > 10000 nM T30082 CA84DP 118558056 IC50 > 10000 nM T30082 C6MHF0 118558060 IC50 > 10000 nM T30082 CB47JV 118558065 IC50 = 16.5 nM T30082 C75WHI 118558069 IC50 = 556 nM T30082 CDRX58 118622604 IC50 = 33100 nM T30082 CP5Z8M 118622610 IC50 = 7900 nM T30082 C7TZ2R 118622611 IC50 = 39700 nM T30082 CRW07P 118622616 IC50 > 40000 nM T30082 CL0N2E 118706720 IC50 = 65320 nM T30082 C8B5TY 118706722 IC50 = 14350 nM T30082 C5K2NA 118706723 IC50 = 12000 nM T30082 CJ36BL 118706724 IC50 = 46760 nM T30082 C15IOS 118708574 IC50 = 34 nM T30082 C53UJX 118708575 IC50 = 55 nM T30082 C9M3EL 118709900 IC50 = 233 nM T30082 CMWO04 118709901 IC50 = 94.2 nM T30082 C39HSZ 118709912 IC50 = 580 nM T30082 CI38GE 118709913 IC50 = 398 nM T30082 CH5V0G 118709914 IC50 = 104 nM T30082 CBP3S5 118709915 IC50 = 2910 nM T30082 CT1J4G 118709916 IC50 = 277 nM T30082 C4IZB0 118709917 Ki = 1940 nM T30082 C7JDT6 118709918 Ki = 2360 nM T30082 CEY60K 118709968 IC50 = 2.06 nM T30082 C8GS0O 118709970 IC50 = 0.006 nM T30082 CAGS07 118709972 IC50 = 14.2 nM T30082 C40GLT 118709974 IC50 = 14.2 nM T30082 CY1BQ6 118710487 IC50 = 33.9 nM T30082 CXT04M 118710490 IC50 = 200.91 nM T30082 C24QHC 118710493 IC50 = 216 nM T30082 CM91OJ 118710494 IC50 = 669 nM T30082 C9FBH6 118710497 IC50 = 534.56 nM T30082 CG3O6T 118710500 IC50 = 4200 nM T30082 CUJ6B1 118710502 IC50 = 56493.7 nM T30082 CBT5N9 118710504 IC50 = 1081.43 nM T30082 CL4F5N 118710507 IC50 = 1200 nM T30082 CG9T7H 118710510 IC50 = 224.91 nM T30082 C58EKO 118710513 IC50 = 1500 nM T30082 CYE24P 118710516 IC50 = 820.35 nM T30082 CLW2E4 118710519 IC50 = 12078.14 nM T30082 C1J0IZ 118711805 Ki = 34.4 nM T30082 C8D5HF 118711806 Ki = 44.3 nM T30082 CLG7K5 118711807 Ki = 39.4 nM T30082 CQB1O3 118711808 Ki = 35.8 nM T30082 C5C3XE 118711809 Ki = 70 nM T30082 C3H2YI 118711810 Ki = 76.1 nM T30082 COUQ50 118711811 Ki = 30.9 nM T30082 COSI80 118711812 Ki = 24.3 nM T30082 CJG10W 118711813 Ki = 30.1 nM T30082 CNH93M 118711814 Ki = 56.1 nM T30082 C2Q8IE 118711815 Ki = 59.6 nM T30082 C3C0QD 118711816 Ki = 42.2 nM T30082 CG62FL 118711817 Ki = 55.2 nM T30082 C9U5SV 118712170 Ki = 50.7 nM T30082 C9KUS7 118712171 Ki = 66.1 nM T30082 CJH4K5 118712172 Ki = 91.1 nM T30082 CB74FU 118712173 Ki = 78.2 nM T30082 CE7GU1 118715259 IC50 = 990 nM T30082 CO2M5F 118715260 IC50 = 2170 nM T30082 CZD84N 118715261 IC50 = 110 nM T30082 C1IVY8 118715262 IC50 = 60 nM T30082 CVN98D 118715709 IC50 = 10470 nM T30082 CG78ML 118715710 IC50 = 8950 nM T30082 CBO21H 118715711 IC50 = 13070 nM T30082 C5JO1E 118715712 IC50 = 22510 nM T30082 CK8MI7 118715713 IC50 = 23210 nM T30082 C5S7WZ 118715714 IC50 = 34140 nM T30082 CN6QV9 118715715 IC50 = 50440 nM T30082 CF0RX8 118715716 IC50 = 64550 nM T30082 C6MD2K 118715717 IC50 = 24630 nM T30082 C57BFX 118715718 IC50 = 5910 nM T30082 C1EJ5Q 118715719 IC50 = 29480 nM T30082 CQ92DR 118715720 IC50 = 44050 nM T30082 CRD9N0 118715721 IC50 = 252960 nM T30082 C6T0HL 118715722 IC50 = 151830 nM T30082 CQS06R 118715723 IC50 = 21940 nM T30082 C31XUV 118715724 IC50 = 76870 nM T30082 C3ZO6M 118715725 IC50 = 162590 nM T30082 CB9DC4 118717254 IC50 = 285.1 nM T30082 C8J0XE 118717257 IC50 = 536.4 nM T30082 CU63FS 118717260 IC50 = 301.1 nM T30082 C59DBS 118717261 IC50 = 426 nM T30082 C64NEL 118717262 IC50 = 390.2 nM T30082 C92IKP 118717263 IC50 = 954.2 nM T30082 CP6G8O 118717405 IC50 = 98.2 nM T30082 C6MIQ1 118717407 IC50 = 325 nM T30082 CXSB36 118717408 IC50 = 92.6 nM T30082 C0D5SZ 118717423 IC50 = 153 nM T30082 C8T3EK 118717426 IC50 = 159 nM T30082 CRV1X2 118717427 IC50 = 306 nM T30082 COH5K8 118717428 IC50 = 149 nM T30082 CKG36J 118717429 IC50 = 187 nM T30082 C7YW9D 118717430 IC50 = 526 nM T30082 C4D5RK 118717431 IC50 = 203 nM T30082 CY0MZ9 118717432 IC50 = 116 nM T30082 C9TX5Y 118717434 IC50 = 153 nM T30082 CUZB16 118719407 IC50 = 17.5 nM T30082 CKMB24 118719408 IC50 = 431 nM T30082 CLE2S7 118720934 IC50 = 6.7 nM T30082 C23AHU 118720935 IC50 = 18.3 nM T30082 CJWC73 118720936 IC50 = 21.1 nM T30082 CTZ2G4 118720937 IC50 = 12110 nM T30082 CCSQ94 118721626 IC50 = 6150 nM T30082 CL7JH8 118721627 IC50 = 103 nM T30082 CK2G3V 118721628 IC50 = 651 nM T30082 CU83LO 118721629 IC50 = 348 nM T30082 CJ3S7L 118721630 IC50 = 1370 nM T30082 C4F0TD 118721871 IC50 = 809 nM T30082 C5MR9S 118721872 IC50 = 3.21 nM T30082 CK85GL 118721873 IC50 = 8.94 nM T30082 CRTA65 118721874 IC50 = 96.1 nM T30082 C6HM0O 118721875 IC50 = 38 nM T30082 C7S9ID 118724460 IC50 = 35120 nM T30082 CO4Q6T 118724461 IC50 = 6300 nM T30082 CHX5E4 118724846 IC50 = 160 nM T30082 C5P3GX 118725584 IC50 = 22000 nM T30082 C0J4XP 118729282 IC50 = 361 nM T30082 C6C9AP 118729283 IC50 = 1831 nM T30082 C6J2RL 118729285 IC50 = 997 nM T30082 C0QN3S 118729287 IC50 = 860 nM T30082 C6PQI9 118729291 IC50 = 525 nM T30082 CF1Z7N 118729293 IC50 = 1992 nM T30082 CYGE08 118729295 IC50 = 625 nM T30082 C68JAH 118729297 IC50 = 644 nM T30082 C4BC2P 118729300 IC50 = 537 nM T30082 CA06HC 118729302 IC50 = 1189 nM T30082 C6CVH3 118729304 IC50 = 1303 nM T30082 C4ZQC8 118729306 IC50 = 1044 nM T30082 C0M3VK 118729722 IC50 > 100 ug.mL-1 T30082 CBD8C5 118729723 IC50 > 100 ug.mL-1 T30082 CTX3W2 118729724 IC50 > 100 ug.mL-1 T30082 CP4D5Q 118729725 IC50 > 100 ug.mL-1 T30082 C0EA2W 118729726 IC50 > 100 ug.mL-1 T30082 CA2P3M 118729727 IC50 > 100 ug.mL-1 T30082 CUC21I 118729728 IC50 > 100 ug.mL-1 T30082 CWU09Y 118729729 IC50 > 100 ug.mL-1 T30082 CLV56Y 118729730 IC50 > 100 ug.mL-1 T30082 C8N5EQ 118729731 IC50 > 100 ug.mL-1 T30082 CH3C4J 118729732 IC50 > 100 ug.mL-1 T30082 CH6P8C 118730042 IC50 = 6.9 nM T30082 CYX21N 118730043 IC50 = 21.6 nM T30082 CJXD41 118730046 IC50 = 17.3 nM T30082 CF73RH 118730047 IC50 = 32.5 nM T30082 CXOA52 118730192 IC50 = 8400 nM T30082 C27ZWI 118730193 IC50 = 15400 nM T30082 CEQ56Z 118730194 IC50 = 4900 nM T30082 C3D6VY 118730195 IC50 = 4600 nM T30082 CJ2P9D 118730196 IC50 = 9600 nM T30082 CI2X8N 118730197 IC50 = 13600 nM T30082 C07TJO 118732687 IC50 = 283.8 nM T30082 CFN57B 118732688 IC50 = 535 nM T30082 C1UWN7 118732689 IC50 = 215.3 nM T30082 C2LJX1 118732690 IC50 = 23.5 nM T30082 C1GS6P 118732691 IC50 = 143.7 nM T30082 CS73OE 118732692 IC50 = 226.5 nM T30082 C62UPS 118732693 IC50 = 453.3 nM T30082 C8BR3S 118733323 IC50 = 202 nM T30082 CFV4Y2 118733324 IC50 = 2105 nM T30082 CRW76M 118733325 IC50 = 303 nM T30082 C9LR2K 118733326 IC50 = 496 nM T30082 CZ83RP 118733328 IC50 = 168 nM T30082 CAI74Z 118733329 IC50 = 941 nM T30082 CKJ80D 118733330 IC50 = 329 nM T30082 CB0M8K 118733331 IC50 = 545 nM T30082 C3CT9I 118733333 IC50 = 268 nM T30082 CTE32X 118733334 IC50 = 3167 nM T30082 CM9L7X 118733337 IC50 = 258 nM T30082 CK43MC 118733338 IC50 = 1596 nM T30082 C6C9XZ 118733339 IC50 = 381 nM T30082 C42RNX 118733340 IC50 = 578 nM T30082 C64CNI 118733342 IC50 = 160 nM T30082 CJ04YT 118733343 IC50 = 2008 nM T30082 CY04NG 118733344 IC50 = 651 nM T30082 CTF87X 118733345 IC50 = 686 nM T30082 CMD97K 118733386 IC50 = 270 nM T30082 CFW53X 118734508 IC50 = 937 nM T30082 CK0WB3 118734509 IC50 = 577 nM T30082 CW3CK1 118734510 IC50 = 69 nM T30082 C2L5JR 118734511 IC50 = 57 nM T30082 CAR91V 118734513 IC50 = 118 nM T30082 C05CSD 118734514 IC50 = 222 nM T30082 CUP7C8 118734515 IC50 = 321 nM T30082 CU4P3W 118734516 IC50 = 8.5 nM T30082 C7QP3J 118734517 IC50 = 45 nM T30082 CVA2J9 118734518 IC50 = 121 nM T30082 C67BGC 118734519 IC50 = 24 nM T30082 CXV5D1 118734521 IC50 = 1030 nM T30082 CLJ19G 118734523 IC50 = 2720 nM T30082 CNB83Q 118734712 IC50 = 24.37 nM T30082 CX80VO 118734713 IC50 = 16.11 nM T30082 C87YTM 118736706 IC50 > 5000 nM T30082 C4CTX6 118736714 IC50 = 2800 nM T30082 CMB54K 118736716 IC50 = 1900 nM T30082 COS59D 118736718 IC50 = 2400 nM T30082 CIB78Z 118736720 IC50 = 700 nM T30082 C2PO6M 118736722 IC50 = 300 nM T30082 C1K2NC 122177803 IC50 = 200 nM T30082 CD4EV0 122177806 IC50 = 950 nM T30082 C4U3BA 122177807 IC50 = 1360 nM T30082 CM1K9Y 122177808 IC50 = 500 nM T30082 CONH53 122177809 IC50 = 80 nM T30082 C6ZP1L 122177815 IC50 = 430 nM T30082 CV6A1K 122177818 IC50 = 900 nM T30082 C2LZ6M 122177820 IC50 = 250 nM T30082 C39GPY 122177822 IC50 = 2000 nM T30082 CT0UG6 122178952 IC50 = 37200 nM T30082 CS9ME8 122178953 IC50 = 25400 nM T30082 CCS52I 122178955 IC50 = 26400 nM T30082 C8ZYI3 122178959 IC50 = 9800 nM T30082 CPKX90 122179856 Ki = 0.0056 nM T30082 CQ2P5O 122179857 Ki = 0.0045 nM T30082 CVB9C4 122179858 Ki = 0.0051 nM T30082 CO6QP7 122179859 Ki = 0.0229 nM T30082 CP01MN 122179860 Ki = 0.0105 nM T30082 CJG71H 122179861 Ki = 0.0081 nM T30082 C0YHI7 122180159 IC50 > 30000 nM T30082 C5K0RY 122180160 IC50 = 10670 nM T30082 C71TKE 122180161 IC50 = 9980 nM T30082 C9QKP3 122180162 IC50 = 1690 nM T30082 CQL13W 122180163 IC50 > 30000 nM T30082 CMR72I 122180164 IC50 = 220 nM T30082 CM5R7F 122180400 IC50 = 1000 nM T30082 C6PTD5 122180404 IC50 = 790 nM T30082 C1X9KB 122180406 IC50 = 300 nM T30082 CMC26Y 122180416 IC50 = 340 nM T30082 C8UIY9 122180417 IC50 = 440 nM T30082 CEJ8S0 122180431 IC50 = 950 nM T30082 C6XI7W 122180432 IC50 = 500 nM T30082 C4OGF8 122180435 IC50 = 910 nM T30082 CJK24Z 122180436 IC50 = 450 nM T30082 CF80GW 122180447 IC50 = 1000 nM T30082 C3ZJF5 122180450 IC50 = 6000 nM T30082 C5LT1G 122180455 IC50 = 8500 nM T30082 CTO9N3 122180457 IC50 = 3900 nM T30082 CKM1E7 122180462 IC50 = 120 nM T30082 CMD2B6 122180465 IC50 = 330 nM T30082 CR8CT0 122183172 IC50 = 4977.37 nM T30082 C2N5MF 122183198 IC50 = 15135.61 nM T30082 C9YTW0 122183199 IC50 = 550000 nM T30082 C51NGK 122183200 IC50 = 3198.9 nM T30082 CIXT08 122183201 IC50 = 879.02 nM T30082 CMC64Z 122183202 IC50 = 2157.74 nM T30082 CVY73R 122183203 IC50 = 510.5 nM T30082 C3BWH1 122183695 IC50 = 62000 nM T30082 CGX20O 122183703 IC50 = 7830 nM T30082 C1ANV4 122184347 IC50 = 1.92 nM T30082 CZ8QL9 122184348 IC50 = 3.46 nM T30082 C3BKN1 122184349 IC50 = 6.46 nM T30082 CPQ19S 122184350 IC50 = 10.1 nM T30082 CG3AN8 122184351 IC50 = 1.48 nM T30082 C7WF3P 122184352 IC50 = 3.66 nM T30082 C8J0OS 122185531 IC50 = 12100 nM T30082 CT2LR8 122185533 IC50 = 19 nM T30082 CFZP30 122185535 IC50 = 295 nM T30082 C3UXJ0 122185537 IC50 = 357 nM T30082 C03AML 122185539 IC50 = 64 nM T30082 CGEY50 122185541 IC50 = 75 nM T30082 C59CJS 122185543 IC50 = 77 nM T30082 CIP98U 122185545 IC50 = 125 nM T30082 CDI8W2 122186374 IC50 > 500000 nM T30082 CK0WP5 122186375 IC50 = 359720 nM T30082 CA7U0N 122186376 IC50 > 500000 nM T30082 CE67WU 122186379 IC50 < 500000 nM T30082 CLTA13 122186382 IC50 = 138230 nM T30082 C8NRX7 122186486 IC50 = 9520 nM T30082 CMCJ76 122186487 IC50 = 133230 nM T30082 C8KFR9 122186490 IC50 = 412560 nM T30082 CV4EJ3 122186491 IC50 = 6710 nM T30082 CU08GD 122186492 IC50 = 187510 nM T30082 CI7UZ4 122186493 IC50 < 500000 nM T30082 CKYL61 122186494 IC50 = 260630 nM T30082 CDU7H8 122186496 IC50 < 500000 nM T30082 C1T7UF 122186498 IC50 = 310310 nM T30082 C21LZX 122186499 IC50 > 500000 nM T30082 CZ38FY 122186500 IC50 > 500000 nM T30082 CGZ6L3 122186501 IC50 = 161340 nM T30082 C8CGX0 122186502 IC50 = 123770 nM T30082 CD37LR 122186505 IC50 = 251670 nM T30082 CP4V8H 122191089 IC50 = 7 nM T30082 C7OGL4 122191091 IC50 = 130 nM T30082 C73UCL 122191093 IC50 = 4000 nM T30082 CA94EV 122192579 IC50 = 6.05 nM T30082 C3NR8D 122192580 IC50 = 869 nM T30082 CZO2U4 122192581 IC50 = 85.9 nM T30082 CR2SK3 122192582 IC50 = 158 nM T30082 C95SVU 122192583 IC50 = 28.8 nM T30082 C7T4YR 122192584 IC50 = 208 nM T30082 CS8Y3D 122192585 IC50 = 578 nM T30082 CC80JL 122192586 IC50 > 10000 nM T30082 CI7W2A 122192587 IC50 = 16900 nM T30082 CFX26L 122192588 IC50 = 17600 nM T30082 C47INY 122192589 IC50 = 5190 nM T30082 CVZ2M4 122192590 IC50 = 1310 nM T30082 CZX9J6 122192591 IC50 > 10000 nM T30082 C16CXB 122193107 IC50 = 30500 nM T30082 C0Q6AY 122193108 IC50 = 28600 nM T30082 CM8C5G 122193110 IC50 = 4200 nM T30082 CBQW34 122193112 IC50 = 3200 nM T30082 CAXZ47 122193114 IC50 = 3900 nM T30082 C0ASQ2 122193116 IC50 = 3400 nM T30082 CXN7T8 122193118 IC50 = 2700 nM T30082 CDKJ53 122193120 IC50 = 5700 nM T30082 CY6H5T 122193122 IC50 = 22900 nM T30082 C6S7CV 122193124 IC50 = 3300 nM T30082 CL8J3Z 122193126 IC50 = 3800 nM T30082 CZ96MQ 122193128 IC50 = 5100 nM T30082 CCZJ35 122193130 IC50 = 1300 nM T30082 C7N1BE 122193132 IC50 = 260 nM T30082 C0FJ1G 122193134 IC50 = 110 nM T30082 CSU6Q5 122193237 IC50 = 210 nM T30082 CSY2D4 122193239 IC50 = 530 nM T30082 C5VTJ4 122193241 IC50 = 440 nM T30082 C5XAM3 122193243 IC50 = 580 nM T30082 CC7E1R 122194787 IC50 = 4360 nM T30082 CNH49U 122194788 IC50 = 1540 nM T30082 CLG31E 122194789 IC50 = 7210 nM T30082 CLOD26 122194790 IC50 = 13290 nM T30082 CY3EJ9 122194791 IC50 = 6610 nM T30082 CI7Q9F 122194792 IC50 = 6720 nM T30082 C9C7VG 122194793 IC50 = 3480 nM T30082 C2A4ES 122194881 IC50 = 260 nM T30082 CI2K5Z 122194882 IC50 = 210 nM T30082 C1E3LP 122194883 IC50 = 80 nM T30082 C4A8JM 122194884 IC50 = 150 nM T30082 CR79OE 122194885 IC50 = 120 nM T30082 CZ8L9J 122194886 IC50 = 100 nM T30082 CK7B8R 122194887 IC50 = 80 nM T30082 CSNM01 122194888 Ki = 49.5 nM T30082 C5JXL2 122199175 IC50 = 2200 nM T30082 CEX9B4 122199179 IC50 = 800 nM T30082 CPJ2K1 122199184 IC50 = 600 nM T30082 C3N9DJ 122199186 IC50 = 6700 nM T30082 C1T5SW 122199188 IC50 = 90 nM T30082 CJV5B8 122387041 IC50 = 6500 nM T30082 CI89OZ 122387042 IC50 = 7900 nM T30082 CYWM69 122387043 IC50 = 6400 nM T30082 CFVL05 122387044 IC50 = 6700 nM T30082 CFI4B3 122387045 IC50 = 6200 nM T30082 CNS65E 122387046 IC50 = 4600 nM T30082 CR63CD 127024868 IC50 = 9600 nM T30082 CFM21Z 127024869 IC50 = 7100 nM T30082 CO01UP 127025001 IC50 = 1690 nM T30082 CT6H9W 127025002 IC50 = 1820 nM T30082 C2Q8FW 127025129 IC50 = 6900 nM T30082 CAB51G 127025336 IC50 = 3960 nM T30082 CO3NW2 127025337 IC50 = 3860 nM T30082 CHW76D 127025338 IC50 = 940 nM T30082 C06WQV 127025339 IC50 = 1390 nM T30082 CN4S6W 127025340 IC50 = 3710 nM T30082 C35YFW 127025347 IC50 = 3240 nM T30082 CU5Y2J 127025348 IC50 = 1150 nM T30082 CZNG40 127025349 IC50 = 1540 nM T30082 CQ32HN 127025350 IC50 = 3370 nM T30082 C8HT6M 127025617 IC50 = 2040 nM T30082 CH6A2X 127026192 IC50 = 1370 nM T30082 C2MHZ4 127026193 IC50 = 67 nM T30082 C71BST 127026245 IC50 = 6000 nM T30082 C5NE2H 127027141 IC50 = 5980 nM T30082 CB25JK 127027142 IC50 = 6240 nM T30082 CT70GX 127027146 IC50 = 610 nM T30082 C10GNQ 127027345 IC50 = 14900 nM T30082 CDV42T 127027424 IC50 = 420 nM T30082 C6M5VF 127027425 IC50 = 1070 nM T30082 CX4YN3 127027643 IC50 = 545 nM T30082 C4AE0D 127027644 IC50 = 424 nM T30082 CJU4L1 127027645 IC50 = 308 nM T30082 CJWO49 127027646 IC50 = 1685 nM T30082 CD5G9O 127027963 IC50 = 24.4 nM T30082 CBC0Y6 127028241 IC50 = 22000 nM T30082 C6R4EA 127028375 IC50 = 3540 nM T30082 CV5C7L 127028376 IC50 = 6590 nM T30082 C0NC1G 127028377 IC50 = 7710 nM T30082 CTF47Q 127028378 IC50 = 5960 nM T30082 CCO6D4 127028379 IC50 = 6370 nM T30082 CYD20X 127028913 IC50 = 5650 nM T30082 C3DGN9 127029030 IC50 = 5800 nM T30082 C3FHL4 127029354 IC50 = 5100 nM T30082 CWJ80N 127029355 IC50 = 6300 nM T30082 C9RD5O 127029356 IC50 = 5900 nM T30082 C3BOU8 127029357 IC50 = 6200 nM T30082 C2VKL4 127030052 IC50 = 242400 nM T30082 CE38AJ 127030670 Ki = 1.59 nM T30082 CKF5Z8 127030955 IC50 = 115900 nM T30082 CE4NT0 127030969 IC50 = 192800 nM T30082 C2ZG6I 127031021 IC50 = 225800 nM T30082 C8I5HY 127031022 IC50 = 341700 nM T30082 CT5OZ6 127031023 IC50 = 341700 nM T30082 CPQ35S 127031025 IC50 = 253000 nM T30082 CN9LT3 127031026 IC50 = 279300 nM T30082 C4T2KL 127031264 Ki = 0.98 nM T30082 C3LM8V 127031334 IC50 = 327000 nM T30082 CXH61I 127031335 IC50 = 235600 nM T30082 CO3G2W 127031336 IC50 = 242400 nM T30082 CY3LR0 127031540 IC50 = 143400 nM T30082 C2V7ZT 127031605 IC50 = 109900 nM T30082 C9FQ2D 127031606 IC50 = 437000 nM T30082 C74QBW 127031607 IC50 = 143400 nM T30082 C0B7WI 127031608 IC50 = 103800 nM T30082 C8SA4R 127031846 Ki = 0.67 nM T30082 C2ILH1 127031859 Ki = 0.72 nM T30082 C7KP3S 127033012 IC50 = 13500 nM T30082 CNH03L 127033707 Ki = 1.34 nM T30082 C8CN4T 127033708 Ki = 1.22 nM T30082 CO31LF 127033915 IC50 = 852 nM T30082 CHC3Y2 127034174 IC50 = 1610 nM T30082 CF3HK1 127034304 IC50 = 110500 nM T30082 C1C8XD 127034555 Ki = 1.06 nM T30082 CC4J3A 127034556 Ki = 0.45 nM T30082 CO48QN 127034557 Ki = 1.05 nM T30082 CRN4X6 127034558 Ki = 0.83 nM T30082 CTAR42 127034559 Ki = 1.33 nM T30082 C67ZWL 127034560 Ki = 1.74 nM T30082 CY1I9K 127034570 IC50 = 80800 nM T30082 CZ3EV8 127035309 IC50 = 2.56 nM T30082 C7TQI5 127035310 IC50 = 2070 nM T30082 CLXU49 127035580 IC50 = 7500 nM T30082 C4BR3Q 127035581 IC50 > 100000 nM T30082 CFB9V2 127035875 IC50 = 1030 nM T30082 C4HJR5 127036051 IC50 = 32.3 nM T30082 CKUR62 127036052 IC50 = 76.9 nM T30082 C1XE2Y 127036053 IC50 = 323 nM T30082 CF19QE 127036054 IC50 = 993 nM T30082 C07GWU 127036055 IC50 = 44.2 nM T30082 CA3MW8 127036212 IC50 = 416 nM T30082 COZ7S8 127036213 IC50 = 47 nM T30082 CW5MQ7 127036214 IC50 = 63.1 nM T30082 CPY5X2 127036215 IC50 = 15.3 nM T30082 C4JFN8 127036216 IC50 = 10.8 nM T30082 CX85YQ 127036232 IC50 = 7495 nM T30082 CS6ND0 127036233 IC50 = 260 nM T30082 CVO6Y9 127036234 IC50 = 1036 nM T30082 C8RI1S 127036330 IC50 = 5900 nM T30082 C1WLH2 127036472 IC50 = 48.6 nM T30082 C65EVQ 127036864 IC50 = 18000 nM T30082 C0RXJ6 127036990 IC50 = 5100 nM T30082 C2LH5V 127037240 IC50 = 222 nM T30082 CH63BP 127037241 IC50 = 117 nM T30082 CIHE05 127037242 IC50 = 200 nM T30082 CT2E9P 127037371 IC50 > 100000 nM T30082 CGUR83 127037375 IC50 > 100000 nM T30082 C8AYT1 127037384 IC50 = 199 nM T30082 CHR89X 127037869 IC50 = 3290 nM T30082 C0RTX1 127038878 IC50 = 6710 nM T30082 CO81HM 127038907 IC50 = 7080 nM T30082 C4QWS0 127043654 IC50 = 150000 nM T30082 CQZW98 127043697 IC50 = 18.3 nM T30082 CCGN43 127043698 IC50 = 6.92 nM T30082 C7XP8D 127043699 IC50 = 255 nM T30082 CCRX05 127043700 IC50 = 922 nM T30082 C5IQU4 127043705 IC50 = 1044 nM T30082 C09KSX 127043865 IC50 = 3800 nM T30082 CG3DR4 127043866 IC50 = 109 nM T30082 CCWJ60 127043867 IC50 = 88.1 nM T30082 CG20QN 127043868 IC50 = 11.3 nM T30082 C3W8MB 127043871 IC50 = 214 nM T30082 C9M0KG 127043877 IC50 = 47900 nM T30082 CZA3R7 127043878 IC50 = 1175 nM T30082 CX1G8L 127043879 IC50 = 157500 nM T30082 C54WIK 127043880 IC50 = 702 nM T30082 CP72LZ 127044176 IC50 = 21.6 nM T30082 C2VJ7H 127044293 IC50 = 130000 nM T30082 CF9BD1 127044471 IC50 = 500000 nM T30082 C5GVQ3 127044472 IC50 = 280000 nM T30082 CT6YL4 127044473 IC50 = 140000 nM T30082 C7S5KZ 127044474 IC50 = 110000 nM T30082 C9GXL0 127044613 IC50 = 1870000 nM T30082 CXS8Z2 127044620 IC50 = 260000 nM T30082 CS0CG7 127044621 IC50 = 2100 nM T30082 CI21OB 127044622 IC50 = 1300 nM T30082 C3PB5G 127044623 IC50 = 460 nM T30082 CXN83I 127044654 IC50 = 125 nM T30082 C97PFW 127044655 IC50 = 312 nM T30082 CC7W8O 127044656 IC50 = 179 nM T30082 C19MEI 127044657 IC50 = 900 nM T30082 CMU0Q3 127045144 IC50 = 89.9 nM T30082 CZOJ81 127045292 IC50 = 80.5 nM T30082 C37IKG 127045293 IC50 = 390 nM T30082 CH6OJ7 127045440 IC50 = 1670000 nM T30082 CRM56I 127045582 IC50 = 1560000 nM T30082 CRG69P 127045583 IC50 = 770000 nM T30082 CFQD76 127048388 IC50 = 25195 nM T30082 C4RGK8 127048389 IC50 = 11135 nM T30082 C8V2DN 127048404 IC50 = 750 nM T30082 CQ16RS 127048405 IC50 = 234 nM T30082 CY71LG 127048406 IC50 = 3300 nM T30082 C7G9XR 127048438 IC50 = 6440 nM T30082 C89GCD 127048439 IC50 = 30670 nM T30082 CW2B3M 127048716 IC50 = 1010 nM T30082 C6GRN5 127048735 IC50 = 12155 nM T30082 CKEN30 127048749 IC50 = 321 nM T30082 C6JQ2A 127049058 IC50 = 1509 nM T30082 C23EOB 127049071 IC50 = 1450 nM T30082 CU8I7J 127049072 IC50 = 2680 nM T30082 C23YAL 127049073 IC50 = 339 nM T30082 C2BVI5 127049123 IC50 = 4630 nM T30082 CG65ES 127049124 IC50 = 13500 nM T30082 CR39WO 127049125 IC50 = 4940 nM T30082 C7X0IE 127049126 IC50 = 9260 nM T30082 CE9K2R 127049377 Ki = 554 nM T30082 CO2U5B 127049378 IC50 = 34500 nM T30082 CU85GC 127049730 IC50 = 390 nM T30082 CRW64G 127049731 IC50 = 1660 nM T30082 C7HV8R 127050028 IC50 = 1540 nM T30082 CW54QX 127050029 IC50 = 1500 nM T30082 C6H2PG 127050318 Ki = 355 nM T30082 CAC15F 127050319 Ki = 1980 nM T30082 CXB9K4 127050511 IC50 = 3800 nM T30082 CCI4E1 127050512 IC50 = 1540 nM T30082 CZGX21 127050513 IC50 = 3600 nM T30082 CS8X7B 127050845 IC50 = 12220 nM T30082 CRE9O5 127051536 IC50 = 5320 nM T30082 C39VRD 127051623 IC50 = 3560 nM T30082 C5CYS7 127051624 IC50 = 7420 nM T30082 CT6FA8 131735884 IC50 = 24 nM T30082 CCA0Q5 131735886 IC50 = 91 nM T30082 C1CS9I 132278164 IC50 = 1300 nM T30082 CKRT62 132278422 IC50 = 800 nM T30082 C16ZYK 132278810 IC50 = 8800 nM T30082 CZ2JQ4 132427688 IC50 = 6.4 nM T30082 C61DGH 132495293 IC50 = 980 nM T30082 CH2K1V 132495294 IC50 = 6390 nM T30082 CM7PY1 132547201 Ki = 520 nM T30082 C3F4ME 132569621 IC50 = 6600 nM T30082 CY3C9T 132569675 IC50 = 8000 nM T30082 C9KGO6 132941375 IC50 = 2500 nM T30082 C3Y4EV 132941376 IC50 = 410 nM T30082 CN1TO8 132941377 IC50 = 360 nM T30082 CB2I0G 132941378 IC50 = 370 nM T30082 CX59ME 133561407 IC50 > 10000 nM T30082 C0LM3G 133721078 IC50 = 138000 nM T30082 C4YH6G 134129916 IC50 = 5780 nM T30082 CG4X6D 134130069 IC50 = 18.2 nM T30082 CO3IZ2 134130116 IC50 = 43.6 nM T30082 CL2XT1 134130413 IC50 = 9.7 nM T30082 C0EU7L 134130629 IC50 = 8430 nM T30082 C5Z9WG 134131252 IC50 = 12.9 nM T30082 CG5H3O 134131347 IC50 = 6.2 nM T30082 C2M8RI 134131482 IC50 = 1.3 nM T30082 CIB75F 134131888 IC50 = 980 nM T30082 CCJF74 134132255 Ki = 14.9 nM T30082 CVF3T5 134133384 IC50 = 64200 nM T30082 CB31IT 134134606 IC50 = 814 nM T30082 CDKC62 134134800 IC50 = 1800 nM T30082 C9OE5Y 134135942 IC50 = 490 nM T30082 CHB06R 134136355 IC50 = 4870 nM T30082 CP3RN6 134136543 IC50 = 1120 nM T30082 CD87VF 134136742 IC50 = 5430 nM T30082 CK06MI 134136825 IC50 = 113 nM T30082 C7XE0G 134137541 IC50 = 8320 nM T30082 CSA09I 134137557 IC50 = 4100 nM T30082 C97CUD 134137716 IC50 = 9700 nM T30082 CYG95X 134137746 IC50 = 97 nM T30082 CK61OC 134138653 IC50 = 1350 nM T30082 CTQY30 134138725 IC50 = 29800 nM T30082 CJ6AO0 134139236 IC50 = 4670 nM T30082 CM5D2F 134139579 IC50 = 73 nM T30082 CU9Q3K 134140017 IC50 = 33 nM T30082 C0VGT1 134140048 IC50 = 10000 nM T30082 C8R7QN 134140515 IC50 = 1010 nM T30082 C4FV6K 134141546 IC50 = 1590 nM T30082 CC6P0J 134141898 IC50 = 195 nM T30082 CUP09Q 134142596 IC50 = 630 nM T30082 C9L1VS 134142725 IC50 = 2960 nM T30082 CAG1P8 134144470 IC50 = 1930 nM T30082 CC26YJ 134145344 IC50 = 1090 nM T30082 CZVL70 134146128 IC50 = 32 nM T30082 C89RCM 134146339 IC50 = 883 nM T30082 CZM9O4 134146757 IC50 = 5990 nM T30082 CW1U8M 134147085 IC50 = 8050 nM T30082 CH0GE5 134147661 IC50 = 730 nM T30082 CT05QR 134147966 IC50 = 3490 nM T30082 CVX5K1 134147979 IC50 = 20900 nM T30082 C7E3YA 134149382 IC50 = 8730 nM T30082 C4Y5ZX 134150471 IC50 = 990 nM T30082 CJ98WY 134152913 IC50 = 4560 nM T30082 CYL06E 134152970 IC50 = 3180 nM T30082 CA2KR0 134153338 IC50 = 3300 nM T30082 CT51CQ 134153533 IC50 = 12600 nM T30082 C8US3H 134154226 IC50 = 1980 nM T30082 CNKI41 134154307 IC50 = 2270 nM T30082 C62PCY 134154918 IC50 = 1480 nM T30082 C9QXG2 134155279 IC50 = 1500 nM T30082 CJ7Y1Q 134155675 IC50 = 114 nM T30082 CPBJ79 134155988 IC50 = 2120 nM T30082 C59WYV 134156876 IC50 = 3220 nM T30082 C5KP8M 134156967 IC50 = 830 nM T30082 CUD08L 134817200 IC50 = 530 nM T30082 CZQS20 134828069 IC50 = 20.4 nM T30082 CYB5V2 134828071 IC50 = 91.4 nM T30082 CHX5W7 134908214 IC50 > 1000 nM T30082 C1GY2T 135156251 EC50 > 10000 nM T30082 CEW6B4 135401162 IC50 = 0.57 nM T30082 CXS6M1 135410029 Ki = 180000 nM T30082 CN54VQ 135412778 IC50 = 667800 nM T30082 C8L4OT 135423666 IC50 = 560000 nM T30082 CP50IR 135424906 IC50 = 4368 nM T30082 CWN2Q8 135441800 IC50 > 50000 nM T30082 C4NUT8 135451012 IC50 = 158000 nM T30082 C41RCW 135473164 Ki = 130.05 nM T30082 CC9R2P 135494161 IC50 = 25.7 nM T30082 CL5N2B 135514780 IC50 = 4520 nM T30082 C6SMT5 135517369 IC50 = 3.631 nM T30082 CYM54X 135567438 IC50 = 250 nM T30082 CE24VM 135567444 IC50 = 2300 nM T30082 C8TQ1R 135595416 IC50 = 2800 nM T30082 CZYK16 135618695 IC50 = 10600 nM T30082 C5YH3F 135621406 IC50 = 1475 nM T30082 CFA4J2 135789800 IC50 > 1000000 nM T30082 C98KNJ 135846078 IC50 = 3108 nM T30082 C81ITK 135846093 IC50 = 3832 nM T30082 C29JLP 135858649 Ki = 22800 nM T30082 C0D1QM 135971444 IC50 = 25 nM T30082 C8PF1A 135971445 IC50 = 16 nM T30082 C6JSZ5 136044149 Ki = 110000 nM T30082 CY20WZ 136044157 IC50 = 260000 nM T30082 CGA64Y 136046122 IC50 = 260 nM T30082 C8NJ6Z 136046123 IC50 = 260 nM T30082 CID8S7 136046124 IC50 = 77 nM T30082 C98BTL 136046125 IC50 = 163 nM T30082 CE1S7H 136046126 IC50 = 307000 nM T30082 C2LTY0 136056469 Ki = 233800 nM T30082 CQ48ED 136056471 Ki = 1625000 nM T30082 CJ7A2L 136056472 Ki = 1926000 nM T30082 CK5JN3 136056473 Ki = 2671000 nM T30082 C4LD5W 136086812 IC50 = 0.48 nM T30082 C4Y6XF 136087062 IC50 = 930000 nM T30082 C8C3BX 136087063 IC50 = 870000 nM T30082 CQSW91 136110931 IC50 = 387560 nM T30082 CS04YJ 136209720 IC50 = 2620 nM T30082 CZ8UM3 136239360 IC50 = 74210 nM T30082 C4TR7Z 136239361 IC50 = 78410 nM T30082 CU5VF2 136244586 IC50 = 206310 nM T30082 CNG5M3 136254439 IC50 = 121110 nM T30082 CH29ZJ 136254440 IC50 = 99410 nM T30082 CYD96O 136254441 IC50 = 90910 nM T30082 C86MBG 136260466 IC50 = 40780 nM T30082 CKC84W 136260526 IC50 = 115110 nM T30082 CVE2S8 136260527 IC50 = 79210 nM T30082 C1X8GA 136260528 IC50 = 119110 nM T30082 C8BAP5 137125243 IC50 < 500000 nM T30082 C85UJA 137133274 IC50 = 2360000 nM T30082 C9VWS7 137133275 IC50 = 990000 nM T30082 C58TYF 137133276 IC50 = 970000 nM T30082 CJ0N2K 137133277 IC50 = 1660000 nM T30082 CBT58L 137133278 IC50 = 2270000 nM T30082 CV35IS 137133279 IC50 = 2490000 nM T30082 CJ72QK 137349228 IC50 = 18000 nM T30082 C7ENS1 137631375 IC50 > 20000 nM T30082 CEL8Q2 137631614 IC50 = 14480 nM T30082 C14DWB 137631637 IC50 = 44.67 nM T30082 C2RA0B 137631650 Ki = 3750 nM T30082 CGD29T 137632143 IC50 = 25.6 nM T30082 CE8QA2 137632181 IC50 = 41500 nM T30082 C5HM3W 137632322 IC50 > 1000 nM T30082 CW90QT 137632533 IC50 = 1250 nM T30082 CX6YO4 137632785 IC50 > 5000 nM T30082 CG21YK 137632803 IC50 = 33860 nM T30082 C93UQE 137632831 IC50 = 18 nM T30082 CIY0P1 137632867 IC50 = 4990 nM T30082 C8RJV3 137633015 IC50 = 11120 nM T30082 CQE2C5 137633051 IC50 = 4400 nM T30082 C8FSZ4 137633176 IC50 > 5000 nM T30082 C4QGM6 137633221 IC50 = 940800 nM T30082 C0HMJ8 137633296 IC50 = 1265000 nM T30082 CF40OB 137633350 IC50 > 1000 nM T30082 CVK1Z4 137633425 IC50 = 18980 nM T30082 CK96PE 137633659 IC50 > 1000000 nM T30082 CEI0T6 137633782 IC50 = 4500 nM T30082 CMD38V 137633845 IC50 = 44560 nM T30082 CM7C8N 137633872 IC50 = 510 nM T30082 C9QLT1 137633879 IC50 = 7140 nM T30082 CN54DF 137634080 IC50 = 1124000 nM T30082 CUS49Q 137634181 IC50 = 1730 nM T30082 CCF19I 137634197 IC50 = 760 nM T30082 CVK63S 137634258 IC50 = 7300 nM T30082 C0T9ZD 137634437 IC50 = 24350 nM T30082 CN1X3A 137634470 IC50 > 1000000 nM T30082 C64WME 137634575 IC50 = 802400 nM T30082 CXDY28 137634711 IC50 = 7400 nM T30082 CUSI50 137634757 IC50 > 5000 nM T30082 C2LA3S 137634832 IC50 = 692500 nM T30082 CUBL80 137634869 IC50 = 3.8 nM T30082 CH2IJ8 137634974 IC50 = 4400 nM T30082 CU0DK7 137635136 IC50 = 4300 nM T30082 CD97LB 137635324 IC50 = 39500 nM T30082 CJ21RK 137635381 IC50 = 500 nM T30082 C7S9TN 137635450 IC50 = 1500 nM T30082 CF08CP 137635497 IC50 = 5050 nM T30082 CF6EZ1 137635781 IC50 = 47.86 nM T30082 C82ELC 137635812 IC50 = 20000 nM T30082 C1GT8Y 137635839 IC50 = 3180 nM T30082 CZD61R 137636335 IC50 = 6000 nM T30082 CXF9A4 137636368 IC50 = 41160 nM T30082 CQ1A2M 137636675 IC50 = 684500 nM T30082 C0HM8K 137636778 IC50 = 1058000 nM T30082 CB7K6M 137636935 IC50 = 543400 nM T30082 CV8W7S 137637059 IC50 = 7500 nM T30082 C2WBP4 137637064 IC50 = 7600 nM T30082 C1Z3IU 137637132 IC50 = 180000 nM T30082 CKB51U 137637339 IC50 = 169.8 nM T30082 CLY5O3 137637382 IC50 > 1000 nM T30082 C2Z5KH 137637592 IC50 = 8400 nM T30082 CW3QD8 137637614 IC50 = 658100 nM T30082 CZ5WE1 137637732 IC50 = 8600 nM T30082 C0I5RD 137637763 IC50 = 393300 nM T30082 CFP1G9 137637896 IC50 = 41060 nM T30082 CFI74R 137637910 IC50 > 5000 nM T30082 C6ENB8 137637977 IC50 = 253 nM T30082 C98WJS 137638081 IC50 = 2.92 nM T30082 C07FMS 137638163 IC50 = 1400 nM T30082 CPG2L1 137638431 IC50 = 780 nM T30082 C45FCN 137638517 IC50 = 190000 nM T30082 C01REG 137638554 IC50 = 50120 nM T30082 CF61LT 137638602 IC50 > 1000000 nM T30082 CC7E4I 137638765 IC50 = 7900 nM T30082 CR5G9J 137638769 IC50 = 7200 nM T30082 C4AX5H 137639047 IC50 = 280 nM T30082 CB09QC 137639078 IC50 = 59.5 nM T30082 C9TDB1 137639386 IC50 = 54300 nM T30082 C6DJ8C 137639617 IC50 = 1110 nM T30082 C89ELW 137639718 IC50 = 4200 nM T30082 CRG16O 137639776 IC50 = 1940 nM T30082 CJ1L2M 137639795 IC50 = 3470 nM T30082 CPK5O7 137639919 IC50 > 5000 nM T30082 CW2N5X 137640052 IC50 > 1000000 nM T30082 C4OGK1 137640096 IC50 = 60100 nM T30082 CW7SU4 137640211 IC50 > 1000 nM T30082 CWHY60 137640221 IC50 = 6690 nM T30082 C3L9PR 137640392 IC50 = 40900 nM T30082 C9KUP4 137640423 IC50 = 4.1 nM T30082 CHF9K4 137640604 IC50 = 32000 nM T30082 C7EN5K 137640663 IC50 = 3600 nM T30082 C2DL0Q 137640678 IC50 = 907800 nM T30082 CLS48N 137641195 IC50 = 15200 nM T30082 CJ1V3P 137641233 IC50 = 11110 nM T30082 CY5NR3 137641257 IC50 = 7200 nM T30082 CC4LH6 137641676 IC50 = 417500 nM T30082 CID79L 137641724 IC50 = 24300 nM T30082 CJU76G 137641727 IC50 = 847900 nM T30082 CXL6G5 137641793 IC50 = 14920 nM T30082 CGK12U 137641841 IC50 = 49800 nM T30082 CED9V8 137641985 IC50 > 5000 nM T30082 CDY1X7 137641989 IC50 = 9930 nM T30082 CPGJ10 137642279 IC50 = 2100 nM T30082 CW3O6F 137642405 IC50 = 1510 nM T30082 C3EL4I 137642431 IC50 = 7200 nM T30082 CX7W6A 137642769 IC50 = 4120 nM T30082 CO4QH5 137643111 IC50 = 7340 nM T30082 CT72VS 137643173 IC50 > 5000 nM T30082 C2W8LQ 137643289 IC50 > 1000000 nM T30082 C9KW6B 137643589 IC50 = 740400 nM T30082 C15JOE 137643788 IC50 = 4800 nM T30082 C49CZB 137643848 IC50 = 4200 nM T30082 C9B2ZE 137644072 IC50 = 6400 nM T30082 CD6XG9 137644159 IC50 = 559300 nM T30082 C9ON7G 137644242 IC50 = 61300 nM T30082 CM2CG5 137644485 IC50 = 69910 nM T30082 CD1F7M 137644494 IC50 = 398.1 nM T30082 C5OEB2 137644607 IC50 > 5000 nM T30082 C4YGM1 137644680 IC50 > 5000 nM T30082 CM91SH 137644867 IC50 = 1560 nM T30082 C0MR8E 137644941 IC50 = 977400 nM T30082 C7TWP1 137644997 IC50 = 590 nM T30082 CTZ35O 137645112 IC50 = 69.7 nM T30082 CSCI58 137645198 IC50 = 8950 nM T30082 C9A7FR 137645247 IC50 = 1567000 nM T30082 C1DHM4 137645326 IC50 = 20000 nM T30082 CAOM59 137645444 Ki = 480 nM T30082 CDO8S4 137645632 IC50 = 911300 nM T30082 C96IFX 137645996 IC50 > 200000 nM T30082 CC2SY8 137646193 IC50 = 8300 nM T30082 CPV4Z7 137646357 IC50 = 100500 nM T30082 CXI1O3 137646388 IC50 = 80110 nM T30082 CAGB15 137646401 IC50 = 890 nM T30082 CV0I6J 137647059 IC50 = 37140 nM T30082 CV6BN8 137647089 IC50 = 4 nM T30082 CQ65DR 137647157 IC50 = 50000 nM T30082 CIC93M 137647425 IC50 = 5.2 nM T30082 CL45YE 137647453 IC50 = 13520 nM T30082 C9J3XC 137647729 IC50 = 7200 nM T30082 C5MJG7 137647822 IC50 = 600 nM T30082 C0ZXC8 137647877 IC50 = 1900 nM T30082 C7LO8T 137647944 IC50 > 20000 nM T30082 C41KDG 137648030 IC50 = 7000 nM T30082 CEC78J 137648049 IC50 = 3820 nM T30082 CW3NA8 137648072 Ki = 13200 nM T30082 CJP1G6 137648183 IC50 = 5600 nM T30082 CC5R7U 137648202 IC50 = 6500 nM T30082 CX7K8F 137648339 IC50 = 14000 nM T30082 C4V8QP 137648482 IC50 = 79.43 nM T30082 CBPK31 137648694 IC50 = 60100 nM T30082 C07ZJU 137648924 IC50 = 23720 nM T30082 CMRI71 137649149 IC50 > 5000 nM T30082 CW2UK0 137649211 IC50 = 5300 nM T30082 CES37N 137649250 IC50 = 16700 nM T30082 CT5FQ6 137649317 IC50 = 229.08 nM T30082 CY8X5O 137649531 IC50 = 18.6 nM T30082 C30VHY 137649676 IC50 = 45550 nM T30082 CS98UQ 137649760 Ki = 4010 nM T30082 C7Z4MI 137649813 IC50 = 7500 nM T30082 C12HUM 137650006 IC50 = 6300 nM T30082 CBFM14 137650067 IC50 = 760 nM T30082 CZ2UV8 137650231 IC50 = 754700 nM T30082 C9O7WC 137650671 IC50 = 700 nM T30082 C9D7CW 137650681 Ki = 3340 nM T30082 CDJ1Y2 137650757 IC50 = 568000 nM T30082 CJW29P 137650881 IC50 = 1200 nM T30082 CH02SU 137651178 IC50 = 0.8 nM T30082 C3BSX2 137651192 IC50 = 678 nM T30082 C3UOR1 137651930 IC50 = 32300 nM T30082 CH9JL6 137652028 IC50 > 20000 nM T30082 C3WL9S 137652298 IC50 = 3040 nM T30082 CW9HL2 137652394 IC50 = 890 nM T30082 CC84NA 137652409 IC50 = 69800 nM T30082 C2JPE0 137652672 IC50 > 200000 nM T30082 C1KSJ8 137652783 IC50 = 6210 nM T30082 CND46Q 137652826 IC50 = 14 nM T30082 CG8BW0 137652851 IC50 = 1320 nM T30082 CHWO15 137652896 IC50 = 7600 nM T30082 CMP3S2 137652915 IC50 = 22 nM T30082 C9KTQ1 137652924 IC50 = 750 nM T30082 CQJ78X 137653099 IC50 = 1830 nM T30082 CFPV35 137653376 IC50 = 19400 nM T30082 CD72ES 137653447 IC50 = 41 nM T30082 CP56IY 137653547 IC50 = 524700 nM T30082 CSO97E 137653574 IC50 = 8500 nM T30082 CG3V4T 137653648 IC50 = 1000 nM T30082 C6O0AJ 137653712 IC50 = 3900 nM T30082 C1AEU9 137654004 IC50 = 150000 nM T30082 CB1I0V 137654237 IC50 = 23200 nM T30082 C0UNA5 137654399 IC50 = 5700 nM T30082 C70VNE 137654551 IC50 = 5.8 nM T30082 C0LR3F 137654627 IC50 = 8500 nM T30082 C6JHD7 137654714 IC50 = 14200 nM T30082 CO25BH 137654740 IC50 = 2100 nM T30082 CT1PA9 137654741 IC50 = 850 nM T30082 C58UJM 137654765 IC50 = 2650 nM T30082 C4UZ6L 137654824 IC50 > 10000 nM T30082 CR6TQ0 137654845 IC50 > 1000000 nM T30082 CAQ92O 137654935 IC50 = 2500 nM T30082 CP3R6K 137655004 IC50 = 5800 nM T30082 CW4FC3 137655099 IC50 > 1000000 nM T30082 CIOA41 137655228 IC50 = 2.9 nM T30082 C4KEF1 137655308 IC50 = 13700 nM T30082 CI93TJ 137655373 IC50 = 1207000 nM T30082 C41UPX 137655797 IC50 > 20000 nM T30082 CB7K2O 137655861 IC50 = 12240 nM T30082 CCA96J 137655921 IC50 = 2300 nM T30082 CMA9P4 137655981 IC50 = 12500 nM T30082 CXI43M 137656037 IC50 = 1370 nM T30082 CC1FN2 137656258 IC50 = 895800 nM T30082 CCZ16Q 137656649 IC50 = 956700 nM T30082 CXUG63 137657249 Ki = 2660 nM T30082 C4XM2Y 137657255 IC50 > 5000 nM T30082 CA26MD 137657287 IC50 > 5000 nM T30082 C61BAH 137657694 IC50 = 41630 nM T30082 C3RP6K 137657780 IC50 = 233700 nM T30082 CJNL70 137657810 IC50 = 1360 nM T30082 CFM2E4 137657871 IC50 = 2850 nM T30082 CW1R3M 137657950 IC50 = 26300 nM T30082 CQ4AP2 137658025 IC50 = 6600 nM T30082 CJIF10 137658142 IC50 > 200000 nM T30082 CTF5A6 137658160 IC50 = 2200 nM T30082 CU4B0Q 137658210 IC50 = 3000 nM T30082 CT51VW 137658213 IC50 = 7000 nM T30082 C15GDM 137658514 IC50 = 33020 nM T30082 C68UBA 137658599 IC50 = 1382000 nM T30082 CJU20M 137658706 IC50 = 700 nM T30082 CC7V1S 137658749 IC50 = 4120 nM T30082 C7F0UA 137658941 IC50 = 636700 nM T30082 CEV12H 137659101 IC50 = 4000 nM T30082 CXJ37R 137659138 IC50 = 3.6 nM T30082 COL58K 137659202 IC50 = 7200 nM T30082 CSP06U 137659306 IC50 = 6800 nM T30082 C6F8PJ 137659322 IC50 > 200000 nM T30082 C81IGT 137659454 IC50 = 73320 nM T30082 CC65MS 137659483 IC50 = 7300 nM T30082 C25GFJ 137659864 IC50 > 1000 nM T30082 CHT89W 137660284 IC50 = 625600 nM T30082 CBD24K 137660365 IC50 = 3700 nM T30082 C8IW5O 137660695 IC50 > 5000 nM T30082 CT7NV3 137660697 IC50 = 5.8 nM T30082 C1C8EV 137660700 IC50 > 1000000 nM T30082 CH34LO 137660979 IC50 = 2910 nM T30082 CKMC76 137661029 IC50 = 35130 nM T30082 CC5K8A 137661080 IC50 = 36500 nM T30082 C6F7QS 137661135 IC50 > 10000 nM T30082 C31MDX 137661164 IC50 = 8700 nM T30082 C7E2OH 137661175 IC50 > 5000 nM T30082 CU1X9M 137661204 IC50 = 39 nM T30082 C4CXO3 137661358 IC50 = 32100 nM T30082 CUI24O 137661381 IC50 = 27860 nM T30082 C7FL2W 137661647 IC50 = 6400 nM T30082 CQV79Z 137661668 IC50 = 7400 nM T30082 CL1MG8 137661699 IC50 = 37.1 nM T30082 C3PXN5 137662062 IC50 = 63 nM T30082 CIJ43L 137662097 IC50 = 2670 nM T30082 CJA7I0 137662139 IC50 = 144.5 nM T30082 C9J4DH 138320049 IC50 = 13.7 nM T30082 CQH9O1 139048127 IC50 > 200000 nM T30082 CGDR34 139049968 IC50 = 3980 nM T30082 CZE1S7 139050820 IC50 > 200000 nM T30082 CN2P8V 139050822 IC50 > 200000 nM T30082 CUJL86 139600209 IC50 = 300 nM T30082 CU3VY8 141700626 IC50 > 10000 nM T30082 CY20TH 141700627 IC50 > 10000 nM T30082 CC50YG 141700631 IC50 > 10000 nM T30082 CW34MN 142762240 IC50 > 20000 nM T30082 C74BND 142762241 IC50 > 20000 nM T30082 CU7SJ0 145722355 IC50 > 10000 nM T30082 C4U5ZC 145949235 IC50 = 58 nM T30082 CHDG06 145949283 IC50 > 10000 nM T30082 CI14LP 145949343 IC50 = 10700 nM T30082 C80HQW 145949396 IC50 = 10800 nM T30082 C2PHB6 145949685 IC50 = 126160 nM T30082 C6VC7F 145949996 IC50 > 200000 nM T30082 C9L7MQ 145950163 IC50 = 37.1 nM T30082 CG8B1X 145950244 IC50 > 100000 nM T30082 COK76S 145950325 IC50 = 31 nM T30082 C9X0PU 145950356 IC50 > 10000 nM T30082 CN1MF4 145950493 IC50 = 3050 nM T30082 CKW78G 145950498 IC50 = 171 nM T30082 CLWB05 145950638 IC50 = 210 nM T30082 C35CUT 145950652 IC50 = 37.3 nM T30082 C5PV1E 145950808 IC50 > 10000 nM T30082 C4Y8RV 145950861 IC50 > 200000 nM T30082 CN4C6I 145951178 IC50 = 4880 nM T30082 CELC68 145951296 IC50 = 470 nM T30082 CC2SB8 145951301 IC50 > 100000 nM T30082 C81CRX 145951391 IC50 = 4040 nM T30082 CI4BN2 145951445 IC50 > 10000 nM T30082 CQ3NO6 145951544 IC50 > 10000 nM T30082 CM9RQ7 145951733 IC50 > 100000 nM T30082 CSU4Y2 145951896 IC50 = 710 nM T30082 C1S9LW 145952033 IC50 = 35610 nM T30082 CV4SR8 145952080 IC50 > 10000 nM T30082 CCYN75 145952166 IC50 = 314 nM T30082 CI92GM 145952223 IC50 > 10000 nM T30082 C8WI5C 145952287 IC50 = 896 nM T30082 CK3M0V 145952290 IC50 > 100000 nM T30082 CB68TN 145952425 IC50 = 1861 nM T30082 CR4B9U 145952544 IC50 = 893.8 nM T30082 C4G3CL 145952548 IC50 > 10000 nM T30082 C0AS6N 145952571 IC50 = 275 nM T30082 C6VLZ8 145952662 IC50 = 14 nM T30082 CK7GU9 145952684 IC50 = 378.8 nM T30082 CGW92C 145952721 IC50 > 30000 nM T30082 CMLV81 145952779 IC50 = 6 nM T30082 CYL7M4 145953009 Ki = 56200 nM T30082 C2SFL4 145953212 IC50 = 8180 nM T30082 C5U8LK 145953230 IC50 = 6160 nM T30082 CN9RI8 145953235 IC50 > 200000 nM T30082 C5AV0L 145953967 IC50 = 78100 nM T30082 C0SBJ8 145954000 IC50 = 18.1 nM T30082 C7D4YV 145954109 IC50 = 93 nM T30082 CU50YP 145954188 IC50 = 21 nM T30082 C84MEQ 145954259 IC50 = 1160 nM T30082 C9ZPF5 145954333 IC50 = 5280 nM T30082 CN8O5L 145954415 IC50 = 10590 nM T30082 C9W2NS 145954473 IC50 > 10000 nM T30082 CCQ80E 145954570 IC50 = 27 nM T30082 CTY0B2 145954599 IC50 = 28300 nM T30082 CVTW73 145954684 IC50 = 116.5 nM T30082 CTAM08 145954688 IC50 > 200000 nM T30082 CGVH54 145954856 IC50 > 200000 nM T30082 CNR7S9 145955032 IC50 > 10000 nM T30082 CRP68J 145955177 IC50 = 10100 nM T30082 C7I2UC 145955258 IC50 > 10000 nM T30082 CU0NC6 145955344 IC50 > 10000 nM T30082 C7B5AO 145955399 IC50 = 143.5 nM T30082 C2D5NS 145955453 IC50 > 10000 nM T30082 C2F3ZI 145955512 IC50 = 30 nM T30082 C71CVO 145955623 IC50 > 10000 nM T30082 CMAH86 145955942 IC50 = 1990 nM T30082 CYQL50 145956161 IC50 > 100000 nM T30082 CY2QK3 145956411 IC50 = 37 nM T30082 CM73CS 145956435 Ki = 98000 nM T30082 CMYF60 145956446 IC50 = 31200 nM T30082 CKP54F 145956485 IC50 > 10000 nM T30082 C4IFB9 145956542 IC50 > 10000 nM T30082 CRTG06 145956559 IC50 = 23800 nM T30082 CWQA30 145956575 IC50 = 11300 nM T30082 CNIR29 145956699 IC50 = 759 nM T30082 CSF0B8 145956727 IC50 > 10000 nM T30082 CF2U6R 145956901 IC50 > 100000 nM T30082 CE2J1F 145956939 IC50 > 200000 nM T30082 CBU9R8 145957015 IC50 > 10000 nM T30082 C7BY3Q 145957085 IC50 = 29800 nM T30082 CEO35K 145957089 IC50 > 200000 nM T30082 C4BEN0 145957301 IC50 = 11 nM T30082 COR92I 145957306 IC50 = 99700 nM T30082 CKRD81 145957336 IC50 > 100000 nM T30082 CBHP60 145957521 IC50 > 10000 nM T30082 CKHG89 145957626 IC50 = 22.2 nM T30082 CB41ZW 145957838 IC50 = 69.3 nM T30082 CW1M4Y 145958077 IC50 = 153 nM T30082 CDQ1O4 145958078 IC50 > 200000 nM T30082 C52DHU 145958113 IC50 = 290 nM T30082 CHQ28Y 145958255 IC50 = 9267 nM T30082 CG6D8I 145958306 IC50 > 10000 nM T30082 CH91EN 145958390 IC50 = 20 nM T30082 CCBO90 145958532 IC50 > 10000 nM T30082 CLA4O5 145958545 IC50 = 610 nM T30082 CPH63I 145958701 IC50 > 200000 nM T30082 CCI31H 145958806 IC50 = 890 nM T30082 C08BCZ 145958863 IC50 = 2.7 nM T30082 C6Q7RS 145958896 IC50 > 100000 nM T30082 CTCE08 145958953 IC50 = 3170 nM T30082 C4TR8I 145959078 IC50 = 242.4 nM T30082 C7ID9N 145959200 IC50 > 200000 nM T30082 C7E0WG 145959287 IC50 = 648 nM T30082 C03XJK 145959323 IC50 > 100000 nM T30082 CWO5K7 145959402 IC50 = 923 nM T30082 C0PNL7 145959576 IC50 = 77 nM T30082 C6GH4S 145959601 IC50 = 8400 nM T30082 C7MIO8 145959624 IC50 = 1160 nM T30082 CNS69M 145959783 IC50 > 10000 nM T30082 CFUJ38 145959883 IC50 = 31000 nM T30082 C32VGH 145959885 IC50 > 200000 nM T30082 C02SYQ 145960412 IC50 = 9130 nM T30082 C9V2GM 145960915 IC50 = 8750 nM T30082 C9UZ6F 145961178 IC50 = 11260 nM T30082 CY4ZE2 145961216 IC50 = 26430 nM T30082 CY1LJ6 145961657 IC50 = 7170 nM T30082 CN0ZW9 145961697 IC50 = 18550 nM T30082 CTX2U0 145961737 IC50 = 10880 nM T30082 C9TJS7 145961749 IC50 = 10720 nM T30082 C4MZ5A 145962235 IC50 = 8830 nM T30082 C4TWG3 145962435 IC50 = 24260 nM T30082 C4DRA8 145962810 IC50 = 19600 nM T30082 CSK58Z 145962855 IC50 = 25070 nM T30082 CRD76Q 145963428 IC50 = 5850 nM T30082 CB3K5N 145963520 IC50 > 10000 nM T30082 CD6K7P 145963526 IC50 = 8850 nM T30082 CBA90S 145963676 IC50 = 12550 nM T30082 CURY23 145963786 IC50 = 0.02836 nM T30082 C37BNF 145963787 IC50 = 24.1 nM T30082 CTH70Y 145963788 IC50 = 78.1 nM T30082 C85ZOK 145963821 IC50 = 491 nM T30082 C8VFP2 145963831 IC50 = 4.09 nM T30082 CIZ2D6 145964146 IC50 = 2640 nM T30082 CUY37P 145964192 IC50 = 310 nM T30082 C06TOS 145964196 IC50 = 0.01893 nM T30082 C9RC3Y 145964200 IC50 = 217.5 nM T30082 CL8IM7 145964214 IC50 = 51.7 nM T30082 CCX4G7 145964403 IC50 = 66.6 nM T30082 C7O1VM 145964717 IC50 = 557 nM T30082 CG5FA8 145964757 IC50 = 35.4 nM T30082 CSQ6M0 145964974 IC50 = 0.02158 nM T30082 C54FVX 145964991 IC50 = 0.01441 nM T30082 CC65HS 145965070 IC50 = 46.4 nM T30082 CYFQ34 145965187 IC50 = 0.02938 nM T30082 C52IFK 145965199 IC50 = 108.4 nM T30082 CKM36P 145965241 IC50 = 3100 nM T30082 C7AD4Q 145965386 IC50 = 1.62 nM T30082 CO20FK 145965438 IC50 = 0.01352 nM T30082 CQBU40 145965602 IC50 = 0.51 nM T30082 CMED83 145965605 IC50 = 250 nM T30082 CO09TS 145966146 IC50 = 119 nM T30082 CZ20XJ 145967112 IC50 = 74300 nM T30082 CCVM34 145967131 Ki = 1.57 nM T30082 C4RFE9 145967436 IC50 = 7260 nM T30082 CSKD74 145967473 IC50 = 2.25 nM T30082 CIN05D 145968525 IC50 = 1 nM T30082 C4CGL8 145968916 IC50 = 5.31 nM T30082 CR8Z2D 145969616 IC50 = 128.6 nM T30082 CIB0S1 145969836 IC50 = 0.02621 nM T30082 C7NB8L 145970781 IC50 = 30.7 nM T30082 C8IRS3 145970790 IC50 = 5800 nM T30082 CNS36B 145971232 IC50 = 7640 nM T30082 C3YRF4 145971257 IC50 = 154 nM T30082 C48YCZ 145971330 IC50 = 0.02094 nM T30082 CS52IM 145971379 IC50 = 65.2 nM T30082 CS2NH6 145971450 IC50 = 24100 nM T30082 CKP39X 145971650 IC50 = 9500 nM T30082 CR1QB5 145971752 IC50 > 200000 nM T30082 C1EG8L 145971761 IC50 = 1940 nM T30082 C0RV3Z 145972056 IC50 = 194 nM T30082 CG21IX 145972199 IC50 = 20 nM T30082 C10KGM 145972388 IC50 = 2240 nM T30082 CADI36 145972622 IC50 = 3040 nM T30082 CVG37T 145972858 IC50 = 36.7 nM T30082 CMB59C 145972994 IC50 = 2760 nM T30082 CHA90Q 145973001 IC50 = 231 nM T30082 CE9U6I 145973015 IC50 = 74.5 nM T30082 C83WHC 145973363 IC50 = 210 nM T30082 C8X5YT 145973525 IC50 = 5420 nM T30082 CR01XP 145973666 IC50 = 129 nM T30082 CV2I6R 145973676 IC50 = 4630 nM T30082 CJB7U5 145973747 IC50 = 1077 nM T30082 CTQO27 145973774 IC50 = 352 nM T30082 C58FVA 145973851 IC50 = 20 nM T30082 C2NH8U 145974121 IC50 = 2600 nM T30082 CP3W4L 145974148 IC50 = 89.6 nM T30082 C7WRK1 145974265 IC50 = 180 nM T30082 CUD2Z0 145974298 IC50 = 8300 nM T30082 C9KNC3 145974491 IC50 = 94.1 nM T30082 C1KBN7 145974504 IC50 = 0.01415 nM T30082 C2CSU4 145974513 IC50 = 25.3 nM T30082 C8VZ5F 145974561 IC50 > 10000 nM T30082 C4HS3V 145974588 IC50 = 0.01672 nM T30082 CJ51HA 145974740 IC50 = 13.3 nM T30082 CXS48G 145974962 IC50 = 1530 nM T30082 C7O4SQ 145974973 IC50 = 36.9 nM T30082 C80VLM 145975022 IC50 = 21.2 nM T30082 C26ZBO 145975126 IC50 = 8020 nM T30082 CTMD94 145975130 IC50 = 230 nM T30082 CHZS47 145975154 IC50 = 65.3 nM T30082 CU2ES3 145975561 IC50 = 10.6 nM T30082 CI3Y7C 145975862 IC50 = 0.01095 nM T30082 C8JVC1 145976117 IC50 = 83.6 nM T30082 CV23TM 145976599 IC50 = 0.02592 nM T30082 CU1NO6 145976650 IC50 = 194 nM T30082 CEXP52 145976876 IC50 = 10000 nM T30082 CRAM60 145977029 IC50 = 1850 nM T30082 CA7W6L 145977052 IC50 = 2.64 nM T30082 CF4A0B 145977178 IC50 = 7.61 nM T30082 CBFC12 145977206 IC50 = 6500 nM T30082 CEO72I 145977249 IC50 = 16.8 nM T30082 COSM78 145977433 IC50 = 25.9 nM T30082 CL9HU4 145977623 IC50 = 528 nM T30082 CKO6P0 145977734 IC50 = 3240 nM T30082 C2UVJ5 145977785 IC50 = 3220 nM T30082 CYW3U1 145978073 IC50 = 187 nM T30082 CV2TD0 145978096 IC50 = 41.6 nM T30082 CUD60Z 145978446 IC50 = 293 nM T30082 C1VW4Y 145978556 IC50 = 0.01323 nM T30082 C3Y2LQ 145978644 IC50 > 10000 nM T30082 CQ6TB5 145978697 IC50 = 119 nM T30082 CE07DW 145978744 IC50 = 768 nM T30082 CQZ0G5 145978902 IC50 = 2780 nM T30082 CHX28E 145978908 IC50 = 30300 nM T30082 CZG8R6 145979011 IC50 = 0.43 nM T30082 CW60IL 145979077 Ki = 3300 nM T30082 C9RQ7P 145979084 IC50 = 6110 nM T30082 CS1Z8Y 145979110 IC50 = 4450 nM T30082 CQK12J 145979174 IC50 = 210 nM T30082 CGWB38 145979348 Ki = 22000 nM T30082 C5LQG4 145979536 IC50 = 9870 nM T30082 C7XLF0 145979801 IC50 = 1.995 nM T30082 CGQ0M4 145979846 IC50 = 8990 nM T30082 CX2RW9 145979866 IC50 = 1380 nM T30082 C1D9ZU 145979972 IC50 = 450 nM T30082 CGDP36 145980029 IC50 = 38 nM T30082 CX2NZ1 145980207 IC50 = 1053500 nM T30082 C6PL4V 145980390 IC50 = 13182.57 nM T30082 CW93VH 145980588 IC50 = 4130 nM T30082 CU0TA8 145980601 IC50 = 1620 nM T30082 C1DGZ7 145980638 IC50 = 1220 nM T30082 CC87DL 145980687 IC50 = 190000 nM T30082 CUJ1M8 145980963 IC50 = 5990 nM T30082 CB9Q6H 145981331 IC50 = 2540 nM T30082 CU1P0H 145981388 IC50 = 4600 nM T30082 C1MG5U 145981700 IC50 = 3290 nM T30082 C1XO2S 145981726 IC50 = 87000 nM T30082 CSNL80 145981760 IC50 = 53 nM T30082 C8TP1V 145981823 IC50 = 2360 nM T30082 CE84KA 145981976 Ki = 21000 nM T30082 CX3M9J 145981988 IC50 = 1410 nM T30082 C8RN0E 145982001 IC50 = 2.1 nM T30082 CS50XZ 145982212 IC50 = 3810 nM T30082 CLD9H6 145982286 IC50 = 130 nM T30082 C34PMT 145982380 IC50 = 125200 nM T30082 CWNB08 145982383 IC50 = 1850 nM T30082 CHV1O6 145982449 IC50 > 100000 nM T30082 CFNJ87 145982457 Ki = 12 nM T30082 CKA7I4 145982543 IC50 = 14.7 nM T30082 CAC72J 145982690 IC50 = 2510 nM T30082 CT64BU 145982814 IC50 = 21.2 nM T30082 C84TNZ 145982889 IC50 > 20000 nM T30082 CT54WG 145983191 IC50 = 33 nM T30082 CE4T3A 145983200 IC50 = 1536500 nM T30082 CH9LR2 145983572 IC50 > 20000 nM T30082 C1SP7F 145983635 IC50 > 20000 nM T30082 C7VJ1L 145983695 IC50 = 3290 nM T30082 CM58DZ 145983847 IC50 > 20000 nM T30082 C9L7RG 145983881 IC50 > 20000 nM T30082 C1E5AS 145983888 IC50 > 20000 nM T30082 CB2N3J 145983966 IC50 > 20000 nM T30082 CE1V5A 145983982 IC50 > 20000 nM T30082 CD0QU1 145984154 IC50 = 19000 nM T30082 C8VRX7 145984259 IC50 = 29.8 nM T30082 CW4X2T 145984359 IC50 = 580 nM T30082 CBZ68H 145984482 IC50 = 44.1 nM T30082 C5D0TS 145984586 IC50 > 20000 nM T30082 CE9IB8 145984734 IC50 = 32.4 nM T30082 CV2D9R 145985684 IC50 > 20000 nM T30082 CCF75S 145986161 IC50 > 20000 nM T30082 CB4HG1 145986433 IC50 = 14000 nM T30082 CI21CS 145986459 IC50 = 2100 nM T30082 C19IWK 145986527 IC50 = 580 nM T30082 CD73AY 145986601 IC50 = 620 nM T30082 CCWA30 145986676 IC50 = 40900 nM T30082 CS1CL3 145986706 IC50 = 64100 nM T30082 CGLW18 145987198 Ki = 42000 nM T30082 CBG81P 145987259 Ki = 24000 nM T30082 CYWE49 145987379 IC50 = 1780 nM T30082 C21BYI 145987407 IC50 = 41 nM T30082 CVM40C 145987439 IC50 = 2440 nM T30082 CJP7H5 145987783 IC50 = 22 nM T30082 C98DHT 145987800 IC50 = 1640 nM T30082 CA82TF 145987838 IC50 = 370 nM T30082 CCW5B8 145987874 IC50 = 844500 nM T30082 CLGS98 145988032 IC50 = 970 nM T30082 C3M1ZO 145988042 IC50 = 91 nM T30082 CA45JZ 145988111 IC50 = 1071.52 nM T30082 CJ4U7L 145988121 IC50 = 3.6 nM T30082 CD19JI 145988321 IC50 = 110000 nM T30082 C0XTH9 145988322 IC50 = 333500 nM T30082 CPH9Y7 145988351 IC50 > 200000 nM T30082 C6HW9I 145988398 IC50 = 13000 nM T30082 CVD20U 145988532 Ki = 190 nM T30082 CE1S3L 145988691 IC50 = 860 nM T30082 C1XU7P 145988798 Ki = 60 nM T30082 C5H1GC 145988865 IC50 = 3470 nM T30082 CWU85M 145989145 IC50 = 20000 nM T30082 CWJ1R2 145989205 IC50 = 750 nM T30082 C1J2OP 145989221 IC50 = 1140 nM T30082 C2A8MY 145989254 IC50 = 25720 nM T30082 CSRK69 145989340 IC50 = 2220 nM T30082 C4C2IS 145989399 IC50 = 3460 nM T30082 CDIS04 145989520 IC50 = 5920 nM T30082 C6RB3V 145989629 IC50 = 660 nM T30082 C6QRA9 145989946 IC50 = 970 nM T30082 C4OAU8 145989956 Ki = 11 nM T30082 CTJ5L4 145989961 IC50 = 9250 nM T30082 CVBP12 145989988 IC50 = 300 nM T30082 CDZX56 145990032 IC50 = 5430 nM T30082 C2AG8U 145990124 IC50 = 8540 nM T30082 C9NTF8 145990243 IC50 = 7490 nM T30082 CDIV28 145990279 IC50 = 3420 nM T30082 C5XO7R 145990329 IC50 = 5100 nM T30082 CI64XC 145990336 IC50 = 805100 nM T30082 CY08FE 145990357 IC50 = 93000 nM T30082 C63USF 145990366 Ki = 36000 nM T30082 CDBW68 145990442 IC50 = 2440 nM T30082 C4N1WB 145990478 IC50 = 1.778 nM T30082 CGP60E 145990565 IC50 = 320 nM T30082 CR59TZ 145990611 IC50 = 33 nM T30082 CQ4R9F 145990749 IC50 = 2230 nM T30082 CCAM14 145990761 IC50 = 22300 nM T30082 C5QZJ4 145990784 Ki = 11 nM T30082 CYS2G9 145991007 IC50 = 965100 nM T30082 CIN02P 145991091 IC50 = 10000 nM T30082 C49DSK 145991370 IC50 = 4900 nM T30082 C3Y7FC 145991399 IC50 = 2120 nM T30082 CST3I4 145991487 IC50 = 131100 nM T30082 CKQ9N2 145991501 IC50 = 14100 nM T30082 C1ZQ0W 145991508 IC50 = 740 nM T30082 C1TN3A 145991548 IC50 = 482500 nM T30082 CKU1A9 145991587 IC50 = 910 nM T30082 C8KUE6 145991747 IC50 = 310 nM T30082 C9L8FJ 145991954 IC50 = 2010 nM T30082 CR69KG 145992024 IC50 = 6.3 nM T30082 C1O3VK 145992136 IC50 = 657 nM T30082 C84LNF 145992210 Ki = 12000 nM T30082 CB9P8D 145992212 IC50 = 1150 nM T30082 CJVT79 145992302 IC50 = 8700 nM T30082 CCHD89 145992329 IC50 = 1151000 nM T30082 C19GZS 145992418 IC50 = 23 nM T30082 CDI31H 145992535 IC50 = 4720 nM T30082 C1WI3A 145992723 Ki = 39 nM T30082 C7WA5I 145992788 IC50 = 1.25 nM T30082 CJ04DE 145992806 IC50 = 980 nM T30082 CUAI94 145992856 IC50 = 9320 nM T30082 CPBJ68 145992936 IC50 = 3610 nM T30082 CF36AC 145993120 Ki = 57 nM T30082 C1FBD7 145993205 IC50 = 300 nM T30082 C5YMR4 145993208 IC50 = 170 nM T30082 CQ61NL 145993296 IC50 = 10132 nM T30082 CY2N1D 145993326 IC50 = 3690 nM T30082 CUVC73 145993378 IC50 = 880 nM T30082 CK54FE 145993438 IC50 = 870 nM T30082 C30CMY 145993498 Ki = 21 nM T30082 C27FDC 145993580 IC50 = 1460 nM T30082 C7H2UE 145993600 IC50 = 2470 nM T30082 CQ9HB3 145993722 IC50 = 0.95 nM T30082 C3YCQ2 145993796 IC50 = 113000 nM T30082 C14EIW 145993803 IC50 = 7680 nM T30082 CO26LK 145993934 IC50 = 7430 nM T30082 C4V2RJ 145994271 IC50 = 300 nM T30082 CN4WJ8 145994281 IC50 = 3540 nM T30082 CU9M1Y 145994293 IC50 = 1330 nM T30082 C47WEC 146682552 IC50 = 28600 nM T30082 C9N8DY 146684358 IC50 = 8200 nM T30082 C06YAR 153979960 IC50 > 10000 nM T30082 CJ8V4Q 153979967 IC50 = 10500 nM T30082 C5B1RI 153979968 IC50 = 9700 nM T30082 CZ2OW7 153979970 IC50 > 10000 nM T30082 C2H9LT 153979972 IC50 = 9700 nM T30082 CD6EF5 153979973 IC50 > 10000 nM T30082 C15LBY 153979974 IC50 > 10000 nM T30082 CTV4G0 153979975 IC50 > 10000 nM T30082 CS4E3M 153979977 IC50 > 10000 nM T30082 CH6A9F 153979986 IC50 = 9400 nM T30082 CBXN70 153979988 IC50 = 11600 nM T30082 C9L8CY 153979991 IC50 = 17000 nM T30082 C94IGO 155510425 IC50 = 11.4 nM T30082 C4UL5F 155510526 IC50 = 0.000005 nM T30082 CRX53K 155510902 IC50 = 571 nM T30082 C2TRD5 155511051 IC50 = 786 nM T30082 CKZ3G2 155511497 IC50 = 55 nM T30082 CN1L2G 155512563 IC50 > 10000 nM T30082 CRV62E 155512901 IC50 > 30000 nM T30082 C8QOL4 155513096 IC50 = 580 nM T30082 CV2HT0 155513316 IC50 = 18300 nM T30082 CLP7Q5 155513372 IC50 = 1.4 nM T30082 C8S4OV 155513382 IC50 = 4920 nM T30082 CE31CI 155514453 IC50 = 4220 nM T30082 CY0E3D 155514519 IC50 > 15000 nM T30082 C4QTY1 155514573 IC50 = 1050 nM T30082 CS0C1V 155515351 IC50 = 3.162 nM T30082 CR7C0G 155515606 IC50 = 1500 nM T30082 CF7WL3 155516468 IC50 = 0.000005 nM T30082 COIQ70 155516605 IC50 = 7030 nM T30082 CI02NB 155516607 IC50 = 9.5 nM T30082 CR4P3Z 155516698 IC50 = 710 nM T30082 C7RY9D 155516892 IC50 = 955300 nM T30082 COQ0I2 155517103 Ki = 879 nM T30082 C7WQF6 155517133 IC50 = 1110 nM T30082 CX6CD2 155517150 IC50 = 102 nM T30082 C7CN4W 155517273 IC50 = 160 nM T30082 C28AKI 155517345 IC50 = 9100 nM T30082 CFG9A1 155517376 IC50 = 900 nM T30082 CJHG75 155517385 Ki = 60.79 nM T30082 C0DR8X 155517455 IC50 > 10000 nM T30082 C0LR8C 155517675 IC50 = 28.8 nM T30082 CHYM62 155517972 IC50 = 77400 nM T30082 CJ1F7P 155518144 IC50 = 148 nM T30082 C62HKG 155518395 IC50 = 58.6 nM T30082 C6XI0C 155518495 IC50 = 55.2 nM T30082 COR6Z3 155518726 IC50 = 7330 nM T30082 CWA5P2 155518864 IC50 > 10000 nM T30082 CT5X0O 155519170 Ki = 16.7 nM T30082 C0XI2C 155519241 IC50 = 1460 nM T30082 CET82F 155519354 IC50 > 10000 nM T30082 CS8DF4 155519439 IC50 = 319200 nM T30082 CEJ87B 155519446 IC50 = 0.73 nM T30082 CS1J8H 155519504 IC50 = 0.000005 nM T30082 C7V3DK 155520023 Ki = 60.79 nM T30082 CW65KH 155520207 IC50 = 6.9 nM T30082 CAIX71 155520508 IC50 > 10000 nM T30082 CQN90Y 155520574 IC50 > 30000 nM T30082 CZR0D3 155520717 IC50 = 1000 nM T30082 CRHP79 155521220 IC50 = 150.7 nM T30082 CP0E2K 155521356 IC50 = 1400 nM T30082 CJ4YH8 155521746 IC50 = 94.1 nM T30082 CHG5D0 155521756 IC50 = 900 nM T30082 C9AT3Q 155521926 IC50 = 0.0076 nM T30082 CC2U3Z 155522419 IC50 = 1.63 nM T30082 C2ML7G 155522745 IC50 = 5240 nM T30082 CZB0F7 155523100 Ki = 60.79 nM T30082 C5D2CI 155523661 IC50 = 40 nM T30082 CU0E6I 155523688 IC50 = 7.943 nM T30082 C19AXN 155523737 IC50 = 140 nM T30082 CS6IJ2 155524198 IC50 = 4800 nM T30082 C9VWZ8 155524523 IC50 = 1.995 nM T30082 CXKP56 155524590 IC50 = 26000 nM T30082 CTR2K7 155524775 IC50 = 0.000005 nM T30082 CWE2B5 155524877 IC50 = 480 nM T30082 CH24YB 155525250 IC50 = 100 nM T30082 CGMH43 155525252 IC50 = 76 nM T30082 CKA2M3 155526429 IC50 = 1300 nM T30082 CMT9X3 155526434 IC50 = 1.259 nM T30082 C6NU8X 155526479 IC50 = 730 nM T30082 CDY49N 155526514 IC50 = 3.162 nM T30082 CK85TG 155526796 IC50 = 1300 nM T30082 C9ZR4K 155526939 Ki = 121 nM T30082 C68XKW 155527023 IC50 = 961 nM T30082 CR7VW0 155528538 IC50 > 10000 nM T30082 CE98VB 155529070 IC50 = 1.3 nM T30082 C1I5XU 155530592 IC50 = 890 nM T30082 CT80OY 155530802 IC50 = 10 nM T30082 C1V6BO 155531034 IC50 > 10000 nM T30082 CDS6H1 155531048 IC50 = 62800 nM T30082 C9NTV0 155531349 IC50 = 49.8 nM T30082 C29REA 155531374 IC50 = 173.5 nM T30082 C3E5FM 155531627 IC50 = 50 nM T30082 C5JAQ6 155531947 IC50 = 0.000005 nM T30082 CWB5N8 155532073 IC50 = 2880 nM T30082 C15PWD 155532152 IC50 = 1050 nM T30082 CMZ73E 155532354 IC50 = 80 nM T30082 C6XQF3 155532358 IC50 = 1.9 nM T30082 C5QI0C 155532410 IC50 = 195 nM T30082 C3G4ZQ 155532469 IC50 > 10000 nM T30082 CQL91M 155532503 IC50 = 940 nM T30082 C9JR7I 155533287 IC50 = 0.000005 nM T30082 CMKT62 155533705 IC50 = 470 nM T30082 C5MI1Q 155533773 IC50 = 0.000005 nM T30082 C8Q0OL 155533954 IC50 = 2 nM T30082 CYN5O8 155534304 IC50 = 840 nM T30082 C9W7XG 155534725 IC50 > 10000 nM T30082 CLOD29 155535170 IC50 = 0.3 nM T30082 CS5A6Y 155535996 IC50 = 620 nM T30082 CT90DI 155536211 IC50 = 11600 nM T30082 CKI2M0 155536368 IC50 = 31.62 nM T30082 CV6NH2 155536546 IC50 = 37 nM T30082 C6C5NV 155536937 Ki = 128.82 nM T30082 CY4D3B 155537306 IC50 = 12000 nM T30082 C6R7XI 155537540 IC50 = 216 nM T30082 CS3T4R 155537864 IC50 = 100200 nM T30082 CA6EU8 155538194 IC50 = 3200 nM T30082 CM0EN3 155538588 IC50 = 205600 nM T30082 C25CET 155539421 IC50 = 2450 nM T30082 CE8C2T 155539594 IC50 = 38 nM T30082 C4ZNO5 155539655 IC50 = 62 nM T30082 C5WI2G 155539893 IC50 > 10000 nM T30082 C9JWY1 155540039 IC50 = 8810 nM T30082 CRW71X 155540051 IC50 = 20.8 nM T30082 CE07LP 155540490 IC50 = 294900 nM T30082 CVKX83 155540924 IC50 > 10000 nM T30082 CE1UC4 155541278 IC50 > 10000 nM T30082 CI64ZO 155541480 IC50 = 2900 nM T30082 CD38QG 155541705 IC50 = 1280 nM T30082 CB5N3V 155541758 IC50 = 276.4 nM T30082 C1G2SL 155541763 IC50 = 311 nM T30082 C19DHY 155541876 IC50 = 250 nM T30082 C2PA7S 155542132 IC50 > 10000 nM T30082 C3UND5 155542248 IC50 = 1160 nM T30082 C8CM4P 155542748 IC50 = 1040 nM T30082 CMO67L 155543176 IC50 = 293 nM T30082 C3XW6I 155543353 IC50 = 137.9 nM T30082 C8TW0A 155543495 IC50 = 590 nM T30082 CJ51LO 155543560 IC50 = 1230 nM T30082 CSKI49 155543595 IC50 = 60.6 nM T30082 C17JEA 155543947 IC50 = 1600 nM T30082 CH7ZX3 155544057 IC50 = 12800 nM T30082 CXPM24 155544137 IC50 = 680 nM T30082 CM5J6Q 155544388 IC50 = 690 nM T30082 CV4MO2 155544490 IC50 = 1500 nM T30082 CE32TS 155544687 IC50 = 716 nM T30082 CMXY60 155545085 IC50 > 10000 nM T30082 CQ8PR1 155545227 IC50 = 535 nM T30082 C4R2HA 155545413 IC50 = 1380 nM T30082 CM1P3X 155545649 IC50 = 630 nM T30082 C8KG6D 155545651 IC50 = 51 nM T30082 C50OZR 155545842 IC50 = 3700 nM T30082 CV06IU 155545951 IC50 = 870 nM T30082 COW1Z3 155546180 IC50 = 142 nM T30082 C47KJH 155546201 IC50 = 860 nM T30082 CM6QN1 155546316 IC50 > 10000 nM T30082 C7L0ZS 155546416 IC50 = 640 nM T30082 CKV03D 155546472 IC50 = 221200 nM T30082 CBPS95 155546845 IC50 = 3940 nM T30082 CL6BT8 155547036 IC50 = 400 nM T30082 CQ6XV1 155547042 IC50 = 7570 nM T30082 CB6Q3L 155547149 IC50 = 0.000005 nM T30082 CD9I8N 155547289 IC50 = 55.1 nM T30082 C0P4NA 155547328 IC50 = 68000 nM T30082 CXY4B1 155547375 IC50 = 1240 nM T30082 CX32QR 155547425 IC50 = 2.7 nM T30082 CS60BV 155547778 IC50 = 100 nM T30082 CIFX72 155547781 IC50 = 1280 nM T30082 C4TQ5J 155548079 IC50 = 133 nM T30082 C5VMU7 155548207 IC50 = 30.7 nM T30082 CD8JZ5 155548223 IC50 = 2100 nM T30082 C4Q7RL 155548245 IC50 = 609 nM T30082 C91ODF 155548523 IC50 = 780 nM T30082 CP85KA 155548858 IC50 = 5700 nM T30082 CFT71V 155549427 IC50 = 20000 nM T30082 C8TUW1 155549491 IC50 > 10000 nM T30082 CQXA98 155549709 IC50 = 275 nM T30082 CO41UF 155549796 IC50 = 84 nM T30082 C9J6LI 155549946 IC50 = 1090 nM T30082 C94KDL 155550161 IC50 = 120 nM T30082 C0A7KH 155550386 IC50 = 5.15 nM T30082 CRHO43 155550463 IC50 = 370 nM T30082 C2DYJ7 155551094 IC50 = 26.2 nM T30082 C0YWH5 155551190 IC50 = 260.6 nM T30082 CUA97V 155551450 IC50 = 216 nM T30082 CFW85H 155551467 Ki = 60.79 nM T30082 CUCF03 155551499 IC50 = 70 nM T30082 CM2X5O 155551629 IC50 = 2730 nM T30082 CU35OW 155552076 IC50 = 20100 nM T30082 CJXS06 155552844 IC50 = 63.1 nM T30082 CD87VC 155553046 IC50 = 506 nM T30082 CKE52P 155553161 IC50 = 750 nM T30082 CUH25G 155553797 IC50 = 1770 nM T30082 CQ2SG6 155554219 IC50 = 66000 nM T30082 CS54UQ 155554734 IC50 = 6900 nM T30082 C0W3LZ 155554767 IC50 = 62 nM T30082 CFNH83 155554841 IC50 = 4030 nM T30082 C0TYD9 155554864 IC50 = 1120 nM T30082 CFK23R 155555484 IC50 = 1200 nM T30082 C7N1YW 155555576 IC50 = 2300 nM T30082 CFW5U2 155555974 IC50 > 10000 nM T30082 C5EPX2 155556231 IC50 = 520 nM T30082 C9YCT8 155556531 IC50 = 168 nM T30082 CD5L2W 155556671 IC50 = 7230 nM T30082 C0WAR6 155556705 IC50 = 19 nM T30082 C2EA7Q 155556733 IC50 = 1300 nM T30082 C7S5JN 155556840 IC50 = 2600 nM T30082 CIK5O9 155556877 IC50 = 0.000005 nM T30082 CDN6B5 155556926 IC50 = 6.3 nM T30082 COS94B 155556946 IC50 = 830 nM T30082 C7IRE9 155557054 IC50 = 5770 nM T30082 CU1G2L 155557132 IC50 = 398.11 nM T30082 CQ7AC5 155557160 IC50 = 68300 nM T30082 CK5Q9E 155557224 IC50 = 320 nM T30082 CI41HC 155557480 IC50 = 19.95 nM T30082 CVH23J 155557537 IC50 = 1.4 nM T30082 CVF40Y 155557821 IC50 = 120 nM T30082 CS28NH 155557943 IC50 = 7.4 nM T30082 CE7GC0 155557995 IC50 = 84.4 nM T30082 C14DCT 155558235 IC50 = 500 nM T30082 CE8PZ1 155559190 IC50 = 11000 nM T30082 CH4MA0 155559209 IC50 = 770 nM T30082 C82GCI 155559240 IC50 = 76 nM T30082 C08NEP 155559748 IC50 = 71.1 nM T30082 CV7M0E 155559813 IC50 = 94 nM T30082 C75KNY 155560373 IC50 > 30000 nM T30082 C4T7HU 155560397 IC50 = 4.2 nM T30082 C0SQ7I 155560420 IC50 = 1300 nM T30082 CI8UF7 155560617 IC50 = 1300 nM T30082 C2VCE7 155560793 IC50 = 5650 nM T30082 CN5WK3 155560822 IC50 = 1100 nM T30082 CLY7Q6 155560920 IC50 = 4400 nM T30082 C95CBX 155561050 IC50 = 440 nM T30082 CP7I9L 155561118 IC50 > 15000 nM T30082 C15FIN 155561744 IC50 = 6.31 nM T30082 C0A9HJ 155562003 IC50 = 0.8 nM T30082 CQ7T8I 155562037 Ki = 630 nM T30082 CUZ64A 155562266 IC50 = 1300 nM T30082 CXA0M8 155562612 IC50 = 15500 nM T30082 CY95WK 155562857 IC50 > 10000 nM T30082 CYG1A7 155562879 IC50 = 570 nM T30082 CD04KI 155562901 IC50 = 226 nM T30082 CUQY46 155563122 IC50 = 2880 nM T30082 CU6NW2 155563256 IC50 = 29 nM T30082 CO32PX 155563567 IC50 = 2320 nM T30082 CTK04N 155563892 IC50 = 4900 nM T30082 CT85FR 155563905 IC50 = 1380 nM T30082 CK8XJ4 155564792 IC50 > 10000 nM T30082 CY6OR7 155564797 IC50 = 480 nM T30082 C27WPT 155565176 IC50 = 610 nM T30082 C3T1UX 155565221 IC50 = 133 nM T30082 CP9K5Z 155565241 Ki = 60.79 nM T30082 CEI7U4 155565422 IC50 = 0.000005 nM T30082 C0LW9V 155565787 IC50 = 559 nM T30082 C5OTD7 155566135 IC50 = 870.96 nM T30082 C7NJY2 155566392 IC50 = 590 nM T30082 C3FPU7 155566420 IC50 = 2800 nM T30082 CWPL14 155566983 IC50 > 100000 nM T30082 C9R2MS 155567099 IC50 = 980 nM T30082 CNQ18H 155567205 IC50 = 454 nM T30082 CM63EC 155567324 IC50 = 79.43 nM T30082 C9L0DT 155567334 IC50 = 3190 nM T30082 CW3Q7C 155567905 IC50 = 14 nM T30082 C3EPS6 155567920 IC50 = 542 nM T30082 CG3BR0 155567943 IC50 = 68000 nM T30082 CRMO93 155567970 IC50 = 0.008 nM T30082 CR24FZ 155568280 IC50 = 2400 nM T30082 CDQ05E 155568688 IC50 = 2.5 nM T30082 CXC4S3 155568730 IC50 = 0.000005 nM T30082 CQS38V 155568760 IC50 = 650 nM T30082 CUT84A 155568798 IC50 = 400 nM T30082 C13GJW 155568936 IC50 = 2770 nM T30082 C10CZA 155569041 IC50 = 3750 nM T30082 CZGB74 155569334 IC50 = 23.6 nM T30082 CCUZ74 155569448 IC50 = 1340 nM T30082 CXWI82 155569489 IC50 = 1020 nM T30082 CZ6AT4 155569579 IC50 = 47900 nM T30082 CB48KF 10389291 IC50 = 7900 nM T30082 CM6E0Y 118719405 IC50 = 192 nM T30082 C17PYJ 118719406 IC50 = 72.5 nM T30082 CTP68W 12049891 IC50 = 58000 nM T30082 C9I6OH 136056470 Ki = 2303000 nM T30082 CWP36Z 44275205 IC50 = 101000 nM T30082 CVA1H9 44275260 IC50 = 35000 nM T30082 C0DX9E 44275262 IC50 = 99000 nM T30082 CJ0CE6 44275279 IC50 = 80000 nM T30082 CCG9N2 44275296 IC50 = 70000 nM T30082 C6TQB5 44275347 IC50 > 93000 nM T30082 D00AHD 44435223 Ki = 3.5 nM T30082 D00ANJ 1897797 Ki > 100000 nM T30082 D00DKI 10107976 Ki = 0.033 nM T30082 D00MFR 44419695 IC50 = 800 nM T30082 D00PLH 44428832 Ki > 100000 nM T30082 D00RIX 5280443 IC50 = 12 nM T30082 D01EZC 44421938 IC50 = 6250 nM T30082 D01HRG 12884 Ki > 100000 nM T30082 D01HZN 44428835 Ki > 100000 nM T30082 D01MVX 656986 IC50 = 8.8 nM T30082 D01OND 46080 IC50 = 2500 nM T30082 D01VAU 123493 Ki > 100000 nM T30082 D01VCS 44428837 Ki > 100000 nM T30082 D01XGP 123358 Ki > 100000 nM T30082 D02AQM 6918822 IC50 = 1800 nM T30082 D02BDL 8433 Ki > 100000 nM T30082 D02DUJ 65719 IC50 = 150 nM T30082 D02GJG 11043027 Ki > 100000 nM T30082 D02HQS 19377173 Ki > 100000 nM T30082 D02JEZ 5281426 IC50 = 29000000 nM T30082 D02LWX 44419700 IC50 = 4197.59 nM T30082 D02SGJ 19009 IC50 = 1700 nM T30082 D02TLP 11363 Ki > 100000 nM T30082 D02XHM 44421959 IC50 = 388000 nM T30082 D02YSX 197033 IC50 = 45000 nM T30082 D03HZT 89076 Ki > 100000 nM T30082 D03JRX 52945010 IC50 = 1000 nM T30082 D03KMG 726586 IC50 = 392 nM T30082 D03QGB 2766326 IC50 = 3200 nM T30082 D03TPH 87203 Ki > 100000 nM T30082 D03WOS 44381944 IC50 = 68.9 nM T30082 D04AXR 96047 Ki > 100000 nM T30082 D04CDV 44428829 Ki > 100000 nM T30082 D04EXR 251908 Ki > 100000 nM T30082 D04FHZ 9906452 IC50 = 10 nM T30082 D04GTP 23645738 IC50 = 125 nM T30082 D05AVX 60983 Ki > 100000 nM T30082 D05EMT 22574258 Ki > 100000 nM T30082 D05EYA 18946 Ki > 100000 nM T30082 D05GPI 44421960 IC50 = 626000 nM T30082 D05LTW 22574224 Ki > 100000 nM T30082 D05PNO 4135273 Ki > 100000 nM T30082 D05QNR 24827641 IC50 = 16600 nM T30082 D05QOR 5280460 IC50 = 168600 nM T30082 D05QXU 21389 IC50 = 590 nM T30082 D05UJV 52945624 IC50 = 6700 nM T30082 D05VUC 19971657 Ki > 100000 nM T30082 D05XRY 2752926 Ki > 100000 nM T30082 D05ZCX 44435802 Ki > 100000 nM T30082 D05ZUX 44207909 Ki >= 1000 nM T30082 D06FFD 96430 Ki > 100000 nM T30082 D06GYH 16745302 Ki > 100000 nM T30082 D06UXW 107759 IC50 = 5370.32 nM T30082 D06VGD 6724 Ki > 100000 nM T30082 D07CFJ 589576 Ki > 100000 nM T30082 D07EDG 1901244 Ki = 48200 nM T30082 D07RIQ 71028 IC50 > 10000 nM T30082 D07YJG 11351920 Ki = 20 nM T30082 D08AIJ 440735 IC50 = 1663800 nM T30082 D08AOG 90571 Ki > 100000 nM T30082 D08DAE 305 IC50 = 3013006.02 nM T30082 D08LNT 20689 IC50 = 125892.54 nM T30082 D08PWL 52945680 IC50 = 9200 nM T30082 D08TSE 44191463 Ki = 340 nM T30082 D08UET 4939 Ki = 7140 nM T30082 D08UOB 44428840 Ki > 100000 nM T30082 D08XQI 9395 IC50 = 10 nM T30082 D09ALJ 5280805 IC50 = 12 nM T30082 D09BUG 10207 IC50 = 18.37 ug.mL-1 T30082 D09CGV 44419702 IC50 = 984.01 nM T30082 D09GXM 44421953 IC50 = 2820 nM T30082 D09JZY 44245252 IC50 = 75 nM T30082 D09LSR 11437501 Ki > 100000 nM T30082 D09QDC 5420 IC50 = 340000 nM T30082 D09REF 443672 Ki = 430 nM T30082 D09RJH 3632 IC50 = 0.3236 nM T30082 D0A2BE 2780 IC50 = 890 nM T30082 D0AQ3K 44421955 IC50 = 152000 nM T30082 D0AW4P 10868634 Ki > 100000 nM T30082 D0B1TQ 1810509 Ki > 100000 nM T30082 D0B4DT 44421954 IC50 = 10300 nM T30082 D0B6IQ 2301676 Ki = 400000 nM T30082 D0B8YX 75511 Ki > 100000 nM T30082 D0BB2U 2385968 Ki > 100000 nM T30082 D0C0XU 10496398 IC50 = 270 nM T30082 D0C1LI 53378764 IC50 = 380 nM T30082 D0C9AD 277990 Ki > 100000 nM T30082 D0CN8Z 11392969 Ki > 100000 nM T30082 D0D0BI 8371 Ki = 163 nM T30082 D0D2HH 44428834 Ki > 100000 nM T30082 D0D7FN 283893 Ki > 100000 nM T30082 D0DV9Z 44419694 IC50 = 1300 nM T30082 D0DW9J 123072 Ki > 100000 nM T30082 D0E2GV 44191462 Ki = 860 nM T30082 D0E2IG 44428839 Ki > 100000 nM T30082 D0E2LR 9996081 IC50 = 120 nM T30082 D0E3OZ 135412781 IC50 = 640000 nM T30082 D0E4BT 46871648 IC50 = 23200 nM T30082 D0E5ZP 604575 Ki > 100000 nM T30082 D0EK7H 2734793 Ki > 100000 nM T30082 D0ER5C 44419701 IC50 = 1800 nM T30082 D0F3QP 5889042 Ki = 7390 nM T30082 D0F3RN 89801 Ki > 100000 nM T30082 D0F5EJ 11375002 IC50 = 0.253 nM T30082 D0F5VY 94860 Ki = 850 nM T30082 D0FE7A 183782 IC50 = 403 nM T30082 D0FO2B 1923 IC50 > 100 nM T30082 D0G0GZ 19916609 Ki = 9360 nM T30082 D0G2DQ 4669250 Ki > 100000 nM T30082 D0G2WI 10318177 IC50 = 0.4786 nM T30082 D0G3TK 5280863 Ki = 92800 nM T30082 D0G5QX 135565598 IC50 = 167000 nM T30082 D0G5TL 44419706 IC50 = 1896.71 nM T30082 D0G8FT 230710 IC50 = 840 nM T30082 D0H2UG 52946279 IC50 = 1600 nM T30082 D0H3BC 44421943 IC50 = 7780 nM T30082 D0H9UT 277 IC50 = 67000 nM T30082 D0I3XA 6422124 IC50 = 86100 nM T30082 D0J1IX 1238015 IC50 = 7400 nM T30082 D0J3SN 1868 IC50 > 10000 nM T30082 D0JH7C 72810 Ki > 100000 nM T30082 D0JI0H 3542734 Ki > 100000 nM T30082 D0K3YM 704259 Ki = 691000 nM T30082 D0K6OM 44428838 Ki > 100000 nM T30082 D0K6PO 316765 Ki > 100000 nM T30082 D0K8AU 46891060 IC50 = 19700 nM T30082 D0L0ZH 215159 IC50 = 540 nM T30082 D0L1ST 2777298 Ki > 100000 nM T30082 D0L3EE 262319 IC50 = 8000 nM T30082 D0L4MF 44428833 Ki > 100000 nM T30082 D0L4OW 9823294 IC50 = 65 nM T30082 D0L5QJ 11408144 IC50 = 2000 nM T30082 D0L9YJ 44421937 IC50 = 2680 nM T30082 D0LJ2F 11806279 Ki > 100000 nM T30082 D0LL8H 25129141 IC50 = 221000 nM T30082 D0M0BM 10399068 IC50 = 1.8 nM T30082 D0M1CG 10425 IC50 = 2917427.01 nM T30082 D0M2EM 4650 Ki = 955 nM T30082 D0M2LD 1476756 IC50 > 1000000 nM T30082 D0M2TY 10168 IC50 > 10000 nM T30082 D0M2ZD 44428831 Ki > 100000 nM T30082 D0M4IE 9549196 IC50 = 0.4 nM T30082 D0M5NR 3794313 Ki > 100000 nM T30082 D0MB3S 22493 IC50 = 549.54 nM T30082 D0MC3U 24827759 IC50 = 5800 nM T30082 D0MF5Y 5281614 IC50 = 12 nM T30082 D0MI0Q 72378 IC50 = 155000 nM T30082 D0N0HK 73252 Ki = 1670 nM T30082 D0N8YZ 2427416 Ki > 100000 nM T30082 D0N9ZR 1718647 Ki > 100000 nM T30082 D0NJ4G 80771 Ki > 100000 nM T30082 D0NJ5W 10055202 Ki = 0.104 nM T30082 D0O0LU 264734 Ki > 100000 nM T30082 D0O1QB 1338 IC50 = 7.998 nM T30082 D0O2OH 9907847 IC50 = 750 nM T30082 D0O8DZ 44421948 IC50 = 2890 nM T30082 D0O8LK 16066832 IC50 = 908000 nM T30082 D0O9YQ 52941983 IC50 = 100 nM T30082 D0OJ9P 49799304 IC50 > 30000 nM T30082 D0P1IK 44428841 Ki > 100000 nM T30082 D0P3VH 893336 IC50 = 7100 nM T30082 D0P5YS 114734 Ki = 1.7 nM T30082 D0PF7F 9928397 IC50 = 10 nM T30082 D0Q2YJ 6763 Ki > 100000 nM T30082 D0Q3EV 52948017 IC50 = 360 nM T30082 D0S1MC 23643351 IC50 = 18 nM T30082 D0S2DW 9844749 Ki = 21.7 nM T30082 D0S6TW 1845 Ki > 100000 nM T30082 D0SP2O 7054 Ki > 100000 nM T30082 D0T0HH 1140 IC50 = 4900 nM T30082 D0T2RY 9948320 Ki >= 1000 nM T30082 D0T3PW 5281672 IC50 = 12 nM T30082 D0T5XC 31494 Ki > 100000 nM T30082 D0U0BV 44428830 Ki > 100000 nM T30082 D0U1SE 84774 IC50 = 816582.37 nM T30082 D0U3JD 16358 Ki > 100000 nM T30082 D0U9AU 11385845 IC50 > 30000 nM T30082 D0UK5A 76996 Ki > 100000 nM T30082 D0UT1X 101375 Ki > 100000 nM T30082 D0UZ8R 71043 Ki > 100000 nM T30082 D0V9EN 689043 IC50 > 100000 nM T30082 D0V9VJ 4884 IC50 = 340000 nM T30082 D0W9VA 10667 Ki = 320 nM T30082 D0WX6R 3477013 Ki = 903 nM T30082 D0X0ER 344135 Ki > 100000 nM T30082 D0X4EV 19770285 IC50 = 9.333 nM T30082 D0X4HG 10765787 IC50 = 0.3 nM T30082 D0XI4U 5319470 IC50 = 2208 nM T30082 D0XL1R 9976105 IC50 = 10 nM T30082 D0Y0XQ 2779383 Ki > 100000 nM T30082 D0Y6RZ 22574214 Ki > 100000 nM T30082 D0Y7FX 8651 Ki > 100000 nM T30082 D0Y7HG 5281616 IC50 = 12 nM T30082 D0Z1WQ 76915 Ki > 100000 nM T30082 D0Z4OS 46891015 IC50 = 14000 nM T30082 D0Z5KQ 8400 Ki > 100000 nM T30082 D0Z6CZ 5139980 Ki > 100000 nM T30082 D0Z6GG 46891014 IC50 = 8700 nM T30082 D0Z6WU 201563 IC50 = 400 nM T30082 D0Z8HX 16786802 Ki > 100000 nM T30082 D0ZI7F 211174 IC50 = 11800 nM T30082 D0ZL6B 3772674 Ki > 100000 nM T30082 D0ZR2T 2732752 Ki > 100000 nM T30082 D0ZT5C 44428828 Ki > 100000 nM T30082 D0ZY4C 46891059 IC50 = 9800 nM T81386 D05SBO 46220502 Ki = 57 nM T81386 D00UZR 5330286 Ki = 364 nM T81386 D05ADP 160355 Ki = 790 nM T81386 D07DTV 11338033 IC50 < 10 nM T81386 D08MXP 44631912 IC50 = 197 nM T81386 D09OHR 118426108 IC50 = 914 nM T81386 D0CY1B 6420138 Ki = 480 nM T81386 D0DX4J 67409219 IC50 = 22 nM T81386 D0E3TC 44259 IC50 = 3.3 nM T81386 D0LF1U 5287969 Ki = 3 nM T81386 D0P1CV 46191454 IC50 = 138 nM T81386 D0PL7P 24983461 IC50 = 26 nM T81386 D0Q9UX 16718576 IC50 = 7700 nM T81386 D0S5RC 3025986 IC50 = 4 nM T81386 D0W8IY 23643976 IC50 = 20 nM T81386 D00OWF 5280953 IC50 = 720 nM T81386 D00PWQ 3820 IC50 = 64 nM T81386 D01CJE 71561915 Ki = 4 nM T81386 D07QIP 44253187 Ki = 11 nM T81386 D0GQ7L 71618654 IC50 = 2 nM T81386 D0NS6I 10037501 IC50 > 10000 nM T81386 D0Q3VZ 135398522 IC50 = 18000 nM T81386 D0D3PX 46926350 IC50 = 4 nM T81386 D0NV9O 45380979 IC50 = 5 nM T81386 D0T3ME 156422 IC50 > 30000 nM T81386 D0U2TQ 644215 IC50 = 13 nM T81386 C24ESN 2608 IC50 > 20000 nM T81386 CVMO57 95875 IC50 > 10000 nM T81386 CT61QM 403993 IC50 > 20000 nM T81386 CRJ81A 403994 IC50 > 20000 nM T81386 CB9F1O 447961 Ki = 4 nM T81386 CH7R8E 709073 Ki > 10000 nM T81386 C5NQV8 725327 Ki > 10000 nM T81386 C8ZP0G 879999 Ki = 7873 nM T81386 C86LNP 2779952 IC50 > 100000 nM T81386 CHGS79 3551941 IC50 = 1100 nM T81386 C3BW1R 5327669 IC50 = 80 nM T81386 C4VTS3 5327723 IC50 > 20000 nM T81386 CJ23HP 5494414 IC50 = 815 nM T81386 COL0X2 6539296 Ki = 2 nM T81386 CQ57EC 9548013 IC50 > 100000 nM T81386 CVX20F 9842276 IC50 = 110 nM T81386 C5S6CZ 9879529 IC50 = 2200 nM T81386 CA6N0T 9922607 IC50 = 26 nM T81386 C7PU4Z 10224714 IC50 = 272 nM T81386 C2B0IU 10421236 IC50 = 2400 nM T81386 C9OX6N 11150562 Ki = 260 nM T81386 C4VJ9B 11163528 Ki = 640 nM T81386 CEW3G8 11163580 Ki = 2 nM T81386 C63NLO 11198278 Ki = 1200 nM T81386 CZEL89 11199830 Ki = 640 nM T81386 C09UEA 11233090 Ki = 3 nM T81386 C69HPR 11257553 Ki = 0.4 nM T81386 CLM0O6 11266412 Ki = 110 nM T81386 CD06EJ 11266891 Ki = 490 nM T81386 CJ29BF 11268167 Ki > 10000 nM T81386 CEJH42 11285002 IC50 = 1 nM T81386 CZH5V3 11287415 Ki > 10000 nM T81386 C70LZE 11289869 Ki = 32 nM T81386 CJS09E 11346863 Ki > 10000 nM T81386 CB37AW 11381775 Ki = 1000 nM T81386 C2YC6J 11428427 Ki = 1900 nM T81386 CD6CZ3 11451037 Ki = 12000 nM T81386 CZM23R 11510921 Ki = 27 nM T81386 CS3R9X 11515154 IC50 > 1000000 nM T81386 CRO96D 11574520 IC50 = 210 nM T81386 CFS35Q 11581762 IC50 = 160 nM T81386 CPO6F9 11610059 IC50 > 1000000 nM T81386 C0HX8F 11624162 IC50 > 1000000 nM T81386 C0JD4E 11675224 Ki = 2 nM T81386 CS39HP 11748985 IC50 = 129 nM T81386 C9PVU7 12111408 IC50 = 260 nM T81386 CM56TR 13422573 IC50 = 300 nM T81386 CTM06S 16719774 IC50 = 2630 nM T81386 C4V9QD 16760027 IC50 = 3400 nM T81386 CV7L6K 17942760 IC50 < 10000 nM T81386 C7YG1N 24759534 IC50 = 45 nM T81386 CPIG05 24799078 IC50 = 1100 nM T81386 CT4RG0 24800068 IC50 = 4600 nM T81386 CLV9T7 24801182 IC50 = 250 nM T81386 CRF61X 24801183 IC50 = 50 nM T81386 CP4ZJ7 24801184 IC50 = 1000 nM T81386 CCPF50 24801698 IC50 > 10000 nM T81386 CI3A6R 24801700 IC50 = 220 nM T81386 CZ48LS 24825971 IC50 > 10000 nM T81386 CW4CR5 24959532 Ki = 17 nM T81386 CCA1J5 25104564 IC50 = 44 nM T81386 CHU23B 25168304 IC50 = 8000 nM T81386 CE65CO 25169529 IC50 = 4 nM T81386 CI39OW 25190761 IC50 = 43 nM T81386 C6M2HV 25190763 IC50 = 200 nM T81386 CX4Z1H 25195254 IC50 = 97 nM T81386 C6XGC4 44224280 Ki = 22 nM T81386 C6RZB3 44253186 Ki = 26 nM T81386 C0J6RA 44253188 Ki = 43 nM T81386 C5Z0TA 44253321 Ki = 17 nM T81386 C9X6EY 44253323 Ki = 6 nM T81386 CU9PY1 44253324 Ki = 8 nM T81386 C9D6XM 44253325 Ki = 6 nM T81386 COM13F 44253464 Ki = 14 nM T81386 C68AKT 44253465 Ki = 8 nM T81386 CB32LJ 44253466 Ki = 5 nM T81386 CS1L6F 44481738 IC50 = 2.8 nM T81386 CCP2E4 44570694 IC50 > 100000 nM T81386 C3UIL7 44582684 IC50 = 5400 nM T81386 CN4RC3 44582716 IC50 > 100000 nM T81386 CZS9G7 44582745 IC50 = 1220 nM T81386 C9MG0D 44582838 IC50 = 16000 nM T81386 CL7GO1 45140949 Ki = 140 nM T81386 C2QS8N 45140950 Ki = 670 nM T81386 C9XTS8 45140951 Ki = 160 nM T81386 CQ0ZI7 45141513 IC50 > 10000 nM T81386 CQ7W3Y 46182043 Ki > 10000 nM T81386 CQJ1W7 46182661 Ki > 10000 nM T81386 C3G6NU 46233557 Ki > 10000 nM T81386 COH1V8 46233558 Ki > 10000 nM T81386 CRLZ94 46912952 IC50 = 370 nM T81386 C1VA0B 46912953 IC50 = 150 nM T81386 C1PG7E 46912955 IC50 = 180 nM T81386 CK7PM2 46918486 IC50 = 240 nM T81386 CY96TA 46926801 IC50 = 1240 nM T81386 CL4F5G 49770981 IC50 = 9 nM T81386 CNJ7B3 49770984 IC50 = 2.1 nM T81386 CEXD01 49770987 IC50 = 5.5 nM T81386 C9ND6Y 49770989 IC50 = 19 nM T81386 CHT50A 49770990 IC50 = 9.6 nM T81386 C05KZR 49770995 IC50 = 6.5 nM T81386 CQ74TB 49771003 IC50 = 9.5 nM T81386 CMXH67 49793229 IC50 > 1000 nM T81386 C51OQB 49835655 IC50 = 1900 nM T81386 C03YLA 49838820 IC50 = 39 nM T81386 CCL3R5 49867929 IC50 = 1790 nM T81386 CS13TA 50991506 IC50 = 2 nM T81386 CK30ES 51000420 IC50 = 1000 nM T81386 C1E0VF 53373586 IC50 = 3 nM T81386 C9F2XO 53380162 IC50 = 10 nM T81386 C8NA4L 53384644 IC50 > 30000 nM T81386 CUP75Y 54582100 IC50 = 220 nM T81386 CA0B2E 54585955 IC50 = 7400 nM T81386 C9DX3J 56649281 IC50 = 117 nM T81386 C4CO5B 57335322 Ki = 1510 nM T81386 C3U4ZR 57335323 Ki > 5000 nM T81386 CDA92B 57335324 Ki > 5000 nM T81386 C6X5RL 57395269 Ki > 5000 nM T81386 CWQD92 57397039 Ki = 3330 nM T81386 CR3I5F 57418686 IC50 = 4800 nM T81386 CZK86D 57855560 IC50 = 52 nM T81386 CF6K1Y 58857683 IC50 = 7300 nM T81386 C56MAG 59379853 IC50 > 10000 nM T81386 CXJ63M 59603829 IC50 = 35 nM T81386 CQEU96 59603842 IC50 = 12 nM T81386 C5PC2T 60167947 IC50 = 14 nM T81386 C03IZC 66493692 Ki > 5000 nM T81386 CVG53Y 66571226 IC50 = 3 nM T81386 CZYQ85 66575811 IC50 = 4 nM T81386 C7GO4Z 66576054 IC50 = 1 nM T81386 CYM0N6 67002844 IC50 > 5000 nM T81386 CG6L5P 67222084 IC50 = 1 nM T81386 CV63UL 67240318 IC50 > 10000 nM T81386 C9QG3B 67630488 IC50 = 1858 nM T81386 CM9A2L 67635788 IC50 = 3438 nM T81386 CS46OY 67642003 IC50 = 6917 nM T81386 CVZ8G0 68915223 IC50 = 30 nM T81386 C5DGR9 69036886 IC50 = 1582 nM T81386 CSL4T5 70680234 Ki = 7 nM T81386 CD1U9J 70682821 Ki = 140 nM T81386 C4U5YD 70684896 Ki = 154 nM T81386 CC4U6V 70684897 Ki = 176 nM T81386 CS3I8K 70684898 Ki = 314 nM T81386 C3WK5U 70684923 IC50 = 1010 nM T81386 CBU4O2 70687054 Ki = 285 nM T81386 C2SHG8 70689145 Ki = 253 nM T81386 C5R1EV 70691236 Ki = 98 nM T81386 C09PBJ 70691237 Ki = 91 nM T81386 C5RAN0 70695451 Ki = 207 nM T81386 CN8T9F 70695463 IC50 = 450 nM T81386 C91HPI 71300299 Ki = 7 nM T81386 CL4R5D 71561659 Ki = 19 nM T81386 C86GKD 71561913 Ki = 932 nM T81386 CSM7B9 71561914 Ki > 5000 nM T81386 C8PN3W 71561916 Ki = 11 nM T81386 CQT62G 71561917 Ki = 5 nM T81386 CG5T3J 71561918 Ki = 98 nM T81386 C3HTA1 71561919 Ki > 5000 nM T81386 C6GE7F 71562041 Ki = 7 nM T81386 CH9VW7 71562042 Ki = 5 nM T81386 C93WIB 71562043 Ki = 22 nM T81386 CY0D8N 71562044 Ki = 6 nM T81386 CB4S0N 71562045 Ki = 9 nM T81386 C2NX5F 71562046 Ki = 7 nM T81386 C5OI2T 71562165 Ki = 4 nM T81386 CRB2K5 71562166 Ki = 3 nM T81386 CW97GT 71562167 Ki = 4 nM T81386 CS5Z8L 71562168 Ki = 5 nM T81386 CBC07G 71562284 Ki > 5000 nM T81386 CD01NB 71562285 Ki = 134 nM T81386 C1HZY0 71562286 Ki = 245 nM T81386 CGJ1T4 71562393 Ki = 278 nM T81386 C0TXO8 71562394 Ki = 156 nM T81386 C8QZH4 71562395 Ki = 2 nM T81386 CLG0V3 71562396 Ki = 3 nM T81386 CGSD62 71562397 Ki = 5 nM T81386 C46LOH 71562398 Ki = 3 nM T81386 C2QCY3 71562399 Ki = 16 nM T81386 C5WZN0 71562504 Ki = 8 nM T81386 CK1MQ9 71562505 Ki = 66 nM T81386 CB0KT1 71562507 Ki = 6185 nM T81386 CN3I5V 71579075 IC50 = 845 nM T81386 C5PO4A 71579076 IC50 > 5000 nM T81386 CN51OL 71579077 IC50 = 3130 nM T81386 CX08VC 71579159 IC50 = 910 nM T81386 CBME42 71579160 IC50 = 285 nM T81386 CP52LT 71579248 IC50 = 165 nM T81386 CB0PQ8 71579250 IC50 = 100 nM T81386 CF3WN8 71579251 IC50 = 106 nM T81386 CPIV81 71617809 IC50 = 2 nM T81386 CI8M9A 71719747 Ki = 110 nM T81386 CJQ60F 71720363 Ki = 7 nM T81386 CV01AY 72204789 Ki = 3 nM T81386 CSD7E0 72708420 IC50 = 1660 nM T81386 CW2V7I 72708421 IC50 = 875 nM T81386 C5M9QS 74222731 Ki = 19 nM T81386 C03CHP 76309866 Ki = 36 nM T81386 CE28UA 76309867 Ki = 11 nM T81386 CK3U8L 76313579 Ki = 8 nM T81386 CQIE64 76313580 Ki = 715 nM T81386 C3THX8 76313581 Ki = 3 nM T81386 C0J8NK 76313582 Ki = 16 nM T81386 C5DT2Q 76317084 Ki = 35 nM T81386 C0SKF8 76317085 Ki = 11 nM T81386 C7F2HZ 76317086 Ki = 7 nM T81386 C94QAD 76328016 Ki = 14 nM T81386 CI7XK1 76331677 Ki = 95 nM T81386 CI6Y1O 76335286 Ki = 11 nM T81386 C18GLW 76901385 IC50 = 40 nM T81386 C94ZBF 78357764 IC50 = 11 nM T81386 C3LC8N 86579886 IC50 = 360 nM T81386 C8RJW4 86579887 IC50 = 407 nM T81386 C2X5LP 86579888 IC50 = 2840 nM T81386 CK83ON 86579889 IC50 > 10000 nM T81386 C8DO9K 86579890 IC50 > 10000 nM T81386 CT7YP5 86579891 IC50 = 3840 nM T81386 CZ6S4L 86579927 IC50 = 6060 nM T81386 C58XBH 86579928 IC50 = 1490 nM T81386 C54DML 86579929 IC50 = 1457 nM T81386 CGDJ58 86579930 IC50 = 333 nM T81386 CC96QK 86579931 IC50 = 9870 nM T81386 CAHR80 86579932 IC50 > 10000 nM T81386 C45KSN 86579970 IC50 = 332 nM T81386 C8SRA6 86579971 IC50 = 1401 nM T81386 CZBL39 86579972 IC50 = 490 nM T81386 CZU83F 86579973 IC50 = 510 nM T81386 CJYM31 86579974 IC50 > 10000 nM T81386 C5Q3JW 86579975 IC50 = 4577 nM T81386 CL2TD5 86580012 IC50 = 3110 nM T81386 C8W0OF 86580013 IC50 = 5220 nM T81386 CIF02W 86580016 IC50 = 197 nM T81386 C5EZN8 86580017 IC50 = 296 nM T81386 C13WIZ 86580040 IC50 = 517 nM T81386 COR40A 86580041 IC50 = 6432 nM T81386 C72CWY 86580042 IC50 = 8056 nM T81386 CJ0V3Z 86580043 IC50 > 10000 nM T81386 CKG75B 86580044 IC50 = 327 nM T81386 CB5NV8 86580063 IC50 = 682 nM T81386 CKGB12 86580064 IC50 = 1019 nM T81386 C8JS6P 86580065 IC50 = 743 nM T81386 CR63XQ 86580086 IC50 = 652 nM T81386 CJ5OM8 86580089 IC50 = 7774 nM T81386 CJV9P3 86580090 IC50 = 5525 nM T81386 CO7G4Q 86580109 IC50 = 7533 nM T81386 C7MR1D 86580110 IC50 = 7474 nM T81386 CYN3J4 86580112 IC50 = 366 nM T81386 C7R3OE 86580113 IC50 = 7022 nM T81386 C5OHK2 86580114 IC50 = 346 nM T81386 C30XEC 86580130 IC50 = 261 nM T81386 CWJ9B8 86580131 IC50 = 842 nM T81386 C0ABV7 86580132 IC50 > 10000 nM T81386 C0BE9Q 86580133 IC50 = 9802 nM T81386 C6PFY1 86580134 IC50 = 418 nM T81386 C2I9LB 86580135 IC50 = 1149 nM T81386 C1VUC4 86580154 IC50 = 523 nM T81386 C30ZNT 86580155 IC50 > 10000 nM T81386 CRD27T 86580156 IC50 > 10000 nM T81386 C4J0WM 86580157 IC50 > 10000 nM T81386 CNW57H 86580158 IC50 > 10000 nM T81386 C1G9WI 86580174 IC50 > 10000 nM T81386 CHK3A7 86580175 IC50 = 6501 nM T81386 CC8HL6 86580176 IC50 = 1040 nM T81386 C16YGP 86580177 IC50 > 10000 nM T81386 CW46AV 86580178 IC50 = 1020 nM T81386 CFSL83 86580194 IC50 = 813 nM T81386 CU4A0W 86580195 IC50 = 3057 nM T81386 CRNV30 86580196 IC50 = 4137 nM T81386 C8F0PO 86580197 IC50 > 10000 nM T81386 C9Y4KF 86580199 IC50 > 10000 nM T81386 CJ10ZU 86580200 IC50 > 10000 nM T81386 CQ7Y9N 86580201 IC50 > 10000 nM T81386 CR0B4J 86580202 IC50 = 429 nM T81386 CS4EU9 86580203 IC50 = 4100 nM T81386 CKQ63Y 86580204 IC50 = 580 nM T81386 CHQW90 86580205 IC50 = 3320 nM T81386 CJM23C 86580206 IC50 = 254 nM T81386 CKJ27B 86580230 IC50 = 870 nM T81386 CAHD76 86580232 IC50 = 5385 nM T81386 COP52T 86580236 IC50 = 248 nM T81386 C0P9UY 86580237 IC50 = 210 nM T81386 CTCN36 86580238 IC50 = 601 nM T81386 C6B0ZA 86580239 IC50 = 143 nM T81386 CB3PG6 86580240 IC50 = 6937 nM T81386 CW7V0X 86580241 IC50 = 5414 nM T81386 C73QAX 86580265 IC50 = 2387 nM T81386 CZWS49 86580266 IC50 = 186 nM T81386 C61UDC 86580267 IC50 > 10000 nM T81386 CXR3L9 86580268 IC50 > 10000 nM T81386 CP4U0X 86580269 IC50 = 212 nM T81386 C9HZ3I 86580270 IC50 = 163 nM T81386 CZ2VC5 86580295 IC50 = 400 nM T81386 CBT34D 86580296 IC50 = 1180 nM T81386 C23YIR 86580297 IC50 = 3100 nM T81386 CO05MV 86580298 IC50 > 10000 nM T81386 C1U8HT 86580299 IC50 > 10000 nM T81386 CHM1B4 86580300 IC50 = 142 nM T81386 C7PWF8 86580301 IC50 = 170 nM T81386 CM79HL 86580319 IC50 > 10000 nM T81386 CQV08T 86580320 IC50 = 1800 nM T81386 C01TWF 86580321 IC50 = 6430 nM T81386 C6QL3T 86580323 IC50 = 5330 nM T81386 C0GYK1 86765296 IC50 = 820 nM T81386 C4BKA6 89429109 IC50 > 10000 nM T81386 C2FOK4 89494280 IC50 = 7600 nM T81386 C1HW4B 89735655 IC50 = 240 nM T81386 CE5L8V 90388565 IC50 = 5000 nM T81386 CCAN79 90645088 IC50 > 10000 nM T81386 CE5M0Z 90645089 IC50 > 10000 nM T81386 C59YRN 90656363 IC50 = 2100 nM T81386 C8LZ3U 90656364 IC50 = 1130 nM T81386 COR92X 90656365 IC50 = 1450 nM T81386 CR8F6G 90656366 IC50 = 3170 nM T81386 C8MPU9 90656367 IC50 = 5240 nM T81386 CVP80S 90765738 IC50 = 800 nM T81386 C0IDT2 91754660 IC50 = 627 nM T81386 CI06RS 91938075 IC50 = 226 nM T81386 CP5L9U 118025540 IC50 = 834 nM T81386 CRNU12 121488167 IC50 = 19 nM T81386 C9MIL3 122188249 IC50 = 96 nM T81386 C53AYQ 122188250 IC50 > 10000 nM T81386 CZO41H 122188251 IC50 > 10000 nM T81386 CLW25J 122188252 IC50 = 291 nM T81386 C23PIE 122188253 IC50 > 10000 nM T81386 CE41KZ 122188254 IC50 > 10000 nM T81386 CHQT85 122188255 IC50 > 10000 nM T81386 CLAD59 122188256 IC50 = 201 nM T81386 CI0W3V 122188257 IC50 > 10000 nM T81386 C3BXR2 122188258 IC50 > 10000 nM T81386 C67GYV 122188259 IC50 > 10000 nM T81386 CE81FB 122188260 IC50 > 10000 nM T81386 CG8VX5 122188261 IC50 > 10000 nM T81386 C9ZKA1 122188262 IC50 > 10000 nM T81386 CQF9I2 122188263 IC50 = 1960 nM T81386 COGF57 122188264 IC50 > 10000 nM T81386 CV8D3O 122188265 IC50 > 10000 nM T81386 CPQ89G 122188266 IC50 = 22 nM T81386 CA4LH8 122188267 IC50 > 10000 nM T81386 CO9LT3 122188268 IC50 = 1064 nM T81386 CRH4E1 122188269 IC50 = 79 nM T81386 CXT3E9 122188270 IC50 = 174 nM T81386 CVEB28 122188271 IC50 = 379 nM T81386 C5E7WK 122188272 IC50 > 10000 nM T81386 CWIR28 122188273 IC50 = 209 nM T81386 CB6I5A 122188274 IC50 > 10000 nM T81386 CA8VH1 122188275 IC50 = 43 nM T81386 C1XAP9 122188276 IC50 = 1165 nM T81386 C0BLT6 122188277 IC50 = 2518 nM T81386 CA6V5M 122188278 IC50 = 6555 nM T81386 CP9H3I 122188279 IC50 = 1144 nM T81386 CV89ZC 122188280 IC50 = 265 nM T81386 C2D5TF 122188281 IC50 = 203 nM T81386 C93VST 122188282 IC50 > 10000 nM T81386 C5FGI7 122188283 IC50 > 10000 nM T81386 CJY4C1 122188365 IC50 > 10000 nM T81386 CC4P7E 122194697 Ki > 10000 nM T81386 CH3BN2 122194698 Ki > 10000 nM T81386 CGD5E3 122194699 Ki > 10000 nM T81386 CYR1F2 122194700 Ki > 10000 nM T81386 C7YMU6 122194701 Ki > 10000 nM T81386 CXW4N0 122596923 IC50 = 20 nM T81386 CC9VH8 123132899 IC50 = 25000 nM T81386 C5ZY7L 124114343 IC50 = 66 nM T81386 C01ANR 124647268 IC50 = 5 nM T81386 CM7Q9A 126534280 Ki > 5000 nM T81386 C0DX6I 126534285 Ki = 220 nM T81386 C7IQB6 126534409 Ki = 1091 nM T81386 CY6AE4 126534479 Ki = 787 nM T81386 CKMP96 126535079 Ki > 5000 nM T81386 CN69YO 126535094 Ki > 5000 nM T81386 CIZC84 126535109 Ki > 5000 nM T81386 CG0LS5 126535118 Ki > 5000 nM T81386 CY3FP0 126535127 Ki = 3570 nM T81386 C0FZD9 126535129 Ki = 1801 nM T81386 C34GOC 126535147 Ki = 258 nM T81386 CIGX71 126535154 Ki > 5000 nM T81386 CQ5I4L 126535157 Ki = 831 nM T81386 CD3L9G 126535189 Ki = 436 nM T81386 C2DY5G 126535576 Ki > 5000 nM T81386 CUJ12L 126535619 Ki = 773 nM T81386 CM5EH6 126535633 Ki = 3717 nM T81386 C2ZRN8 126535648 Ki > 5000 nM T81386 C3LBP8 126559195 Ki > 5000 nM T81386 CGVE64 126559600 Ki = 180 nM T81386 C08IBD 126559601 Ki > 5000 nM T81386 CM8C2D 126559606 Ki = 173 nM T81386 CUS75R 127034835 IC50 = 330 nM T81386 CF46KL 127034840 IC50 = 15600 nM T81386 C4WZ9R 127035029 IC50 = 2570 nM T81386 C93INP 127035031 IC50 = 2450 nM T81386 CO2S5V 127035687 IC50 = 1720 nM T81386 C9L4ZJ 127036079 IC50 = 2020 nM T81386 C26RXZ 127036907 IC50 > 10000 nM T81386 CG2OD6 127037298 IC50 = 780 nM T81386 C9G5SN 127037492 IC50 = 11300 nM T81386 CU26ZC 127050134 IC50 = 1100 nM T81386 C4NA2K 129206291 IC50 = 52 nM T81386 CU6HG7 129206345 IC50 = 28 nM T81386 CV49PB 129206866 IC50 = 47 nM T81386 C5H7CN 129206868 IC50 = 213 nM T81386 CV3NY5 129206869 IC50 = 342 nM T81386 C34SUO 129206884 IC50 = 61 nM T81386 CR27KH 129206982 IC50 = 24 nM T81386 C52VQW 129206983 IC50 = 45 nM T81386 CJE30T 129206987 IC50 = 22 nM T81386 CXR9F7 129206992 IC50 = 42 nM T81386 C4MXG9 129206993 IC50 = 42 nM T81386 C57DPW 129206994 IC50 = 146 nM T81386 C6F0TS 129206995 IC50 = 82 nM T81386 CV15ZN 129206998 IC50 = 159 nM T81386 CK10VD 129206999 IC50 = 40 nM T81386 CIZ6M4 129207000 IC50 = 27 nM T81386 CWS5C4 129245211 IC50 = 1520 nM T81386 CH91ON 129245363 IC50 = 14400 nM T81386 CA2N5C 129245517 IC50 = 1460 nM T81386 C0E2RU 129245526 IC50 = 455 nM T81386 C52PNC 129245623 IC50 = 71 nM T81386 CEYK58 129245795 IC50 = 9190 nM T81386 COR37Y 129245842 IC50 > 20000 nM T81386 CQJK71 129246093 IC50 = 2130 nM T81386 C0GC7N 129246130 IC50 = 240 nM T81386 CG5O2J 129261641 IC50 = 320 nM T81386 C0FM1R 130196825 IC50 = 30.3 nM T81386 C3TS2A 132968992 IC50 = 3 nM T81386 C5IZM6 134139906 IC50 = 88 nM T81386 C1T0RJ 134140050 IC50 = 22 nM T81386 CS7NM9 134140744 IC50 = 8 nM T81386 CJ03VI 134140883 IC50 = 5 nM T81386 CRHT71 134148638 IC50 = 8 nM T81386 CQC7R3 134151342 IC50 = 6 nM T81386 CIE4V9 134153731 IC50 = 8 nM T81386 C80QXH 134813906 IC50 = 16000 nM T81386 CM8DK3 134813913 IC50 = 49 nM T81386 CQP51Y 134814484 IC50 = 1 nM T81386 C3F9OH 135286306 Ki = 286 nM T81386 CN7W4K 135286342 Ki = 141 nM T81386 C1OG7T 135286343 Ki = 1980 nM T81386 CUBM68 135286350 Ki = 2000 nM T81386 C10VEZ 135286352 Ki = 925 nM T81386 C2AS3G 135286354 Ki = 2420 nM T81386 C0ZTC9 135286356 Ki > 5000 nM T81386 CXK89G 135286368 Ki > 5000 nM T81386 CK3DZ2 135286381 Ki = 679 nM T81386 C71CGQ 135286391 Ki = 4990 nM T81386 C89ODF 135286395 Ki = 508 nM T81386 CS32WR 135286434 Ki = 1800 nM T81386 CJW6N5 135296339 Ki = 505 nM T81386 CL67GJ 135296341 Ki > 5000 nM T81386 CDP2F0 135296342 Ki = 1321 nM T81386 CH29JY 135398514 IC50 = 150 nM T81386 CKL5H3 135399637 IC50 = 12400 nM T81386 CS4OW8 135400873 IC50 = 14500 nM T81386 CD2J4G 135401182 IC50 = 26000 nM T81386 CWT5H9 135406876 IC50 = 1500 nM T81386 C4SE6Y 135487452 IC50 = 5600 nM T81386 CBU0J4 135604653 IC50 > 10000 nM T81386 CH90LE 135712510 IC50 = 95 nM T81386 CFU1D4 135744101 IC50 = 280 nM T81386 CST7X3 135870706 IC50 = 15 nM T81386 CF6N2M 135922716 IC50 = 1000 nM T81386 CC23AB 135950281 IC50 = 6100 nM T81386 CAH27O 136219283 IC50 = 10.9 nM T81386 CH0Q2Z 136234577 IC50 = 7400 nM T81386 CV6F4N 136234578 IC50 = 3700 nM T81386 C2G3JY 136234579 IC50 > 10000 nM T81386 C13FTU 136240093 IC50 = 880 nM T81386 CQCW57 136240264 IC50 = 120 nM T81386 C7YR3A 136240265 IC50 = 460 nM T81386 CIE3Q9 136245068 IC50 = 2400 nM T81386 CPU1F9 136245297 IC50 = 31 nM T81386 CBTA26 136247015 IC50 = 940 nM T81386 CZS5B6 136380883 IC50 = 9000 nM T81386 CURA13 136934895 IC50 = 1700 nM T81386 C3BQ7I 136934897 IC50 = 700 nM T81386 CJK96M 136934900 IC50 = 400 nM T81386 C7M5IC 136934901 IC50 = 1900 nM T81386 C7V4XJ 136934903 IC50 = 5600 nM T81386 CZXV40 136934907 IC50 = 300 nM T81386 C8VD6F 136961394 IC50 = 1350 nM T81386 CVHF30 137479140 IC50 = 263 nM T81386 CCX3Q6 137628632 IC50 = 12 nM T81386 CU9O3A 137628639 IC50 = 1.9 nM T81386 CCAZ26 137631656 IC50 = 2000 nM T81386 C3QAV9 137631819 IC50 = 4000 nM T81386 CQ15NR 137631839 IC50 = 200 nM T81386 CHCN75 137632049 IC50 = 280 nM T81386 CEC2D1 137632536 IC50 = 450 nM T81386 C7RAH4 137632779 IC50 < 10000 nM T81386 CDER10 137632999 IC50 = 29 nM T81386 CG8Y0U 137633419 IC50 = 3400 nM T81386 CS9TU2 137633985 IC50 > 10000 nM T81386 CGK3Q6 137634367 IC50 = 1000 nM T81386 C83UKG 137634382 IC50 = 1100 nM T81386 CVD84F 137634496 IC50 = 642 nM T81386 CIUF50 137634527 IC50 > 100000 nM T81386 C6L3HN 137634634 IC50 = 9 nM T81386 CNT7S3 137634818 IC50 > 10000 nM T81386 CCP7X5 137635304 IC50 > 10000 nM T81386 C1AK8X 137635556 IC50 = 620 nM T81386 CV7OF5 137635713 IC50 > 10000 nM T81386 C5QWE1 137635926 IC50 = 800 nM T81386 CJR01E 137636220 IC50 = 38 nM T81386 CKZF46 137638065 IC50 > 10000 nM T81386 CCX37E 137638472 IC50 = 1100 nM T81386 CPO87L 137638509 IC50 = 1100 nM T81386 C7CP2N 137638906 IC50 < 10000 nM T81386 C1UI5N 137638944 IC50 > 10000 nM T81386 CH4RP3 137639514 IC50 = 1000 nM T81386 CX3MQ1 137639546 IC50 = 900 nM T81386 CH3S8N 137640038 IC50 = 2200 nM T81386 CVL0J7 137640533 IC50 = 38000 nM T81386 CXM4G7 137640811 IC50 = 1200 nM T81386 CF83TG 137640934 IC50 = 2100 nM T81386 C42CAG 137641300 IC50 = 160 nM T81386 CWVE69 137643514 IC50 = 2000 nM T81386 CF4Q9X 137643609 IC50 = 350 nM T81386 CYA1F7 137643721 IC50 = 320 nM T81386 C2AG3W 137643887 IC50 > 10000 nM T81386 C4DS3I 137643955 IC50 = 3800 nM T81386 CWIP72 137644498 IC50 = 2800 nM T81386 C23ZPG 137644723 IC50 = 59 nM T81386 CZ4U0W 137644802 IC50 = 1700 nM T81386 CGWC38 137644929 IC50 = 52 nM T81386 CPJ42V 137644974 IC50 > 10000 nM T81386 C8VTQ9 137645650 IC50 = 2200 nM T81386 C7ZOV3 137645947 IC50 = 3700 nM T81386 CB5A4P 137646454 IC50 = 19 nM T81386 CL5NX9 137646497 IC50 = 220 nM T81386 CJ5O2Q 137646673 IC50 > 10000 nM T81386 COU37W 137647335 IC50 = 1300 nM T81386 C21IMP 137647416 IC50 < 10000 nM T81386 C2QB4U 137647543 IC50 = 93 nM T81386 C7O2AW 137647969 IC50 > 10000 nM T81386 C5OJH2 137649318 IC50 > 10000 nM T81386 C9QNG8 137650421 IC50 > 10000 nM T81386 CWG94C 137650926 IC50 > 10000 nM T81386 C8MKN0 137651314 IC50 = 3100 nM T81386 CKL0P4 137651538 IC50 > 10000 nM T81386 CJ14XO 137651668 IC50 = 5600 nM T81386 CH6L2T 137652047 IC50 > 10000 nM T81386 C2B5CY 137652970 IC50 > 10000 nM T81386 C48DVU 137653000 IC50 = 3500 nM T81386 C01URE 137653446 IC50 > 10000 nM T81386 C47FBV 137654225 IC50 > 10000 nM T81386 CA5N2M 137654694 IC50 = 750 nM T81386 CAV71H 137655446 IC50 = 260 nM T81386 C7IU4J 137655848 IC50 = 580 nM T81386 CAJN94 137656331 IC50 = 625 nM T81386 C8TM2H 137656537 IC50 = 570 nM T81386 CP76MY 137656839 IC50 = 700 nM T81386 CQEJ60 137656868 IC50 = 2100 nM T81386 C8IXV2 137657189 IC50 = 11.5 nM T81386 C0JF5D 137657398 IC50 = 310 nM T81386 CJR41C 137657453 IC50 = 27 nM T81386 C84RPJ 137658097 IC50 = 570 nM T81386 C39SEV 137658150 IC50 = 7500 nM T81386 CX8YL9 137658187 IC50 = 220 nM T81386 CTO04D 137658447 IC50 < 10000 nM T81386 C8XFW5 137658772 IC50 = 20 nM T81386 CA2PY1 137658970 IC50 = 600 nM T81386 CJ1TB2 137659239 IC50 > 10000 nM T81386 C3U2OB 137659350 IC50 = 2100 nM T81386 CFL9P1 137659439 IC50 < 10000 nM T81386 C7QM6B 137659788 IC50 < 10000 nM T81386 C6RUD3 137660052 IC50 = 66 nM T81386 C7MI2G 137661183 IC50 > 10000 nM T81386 CDI9V6 137661231 IC50 = 35 nM T81386 CIX41F 137661315 IC50 > 10000 nM T81386 CD0FV8 137661355 IC50 = 8100 nM T81386 C4MJ8D 138105941 IC50 = 25 nM T81386 C5J2WV 138728749 IC50 = 1890 nM T81386 C48TEA 138911336 IC50 = 11 nM T81386 CM07EU 145714274 IC50 > 20000 nM T81386 C3UB5F 145949983 IC50 > 30000 nM T81386 CZ5J1W 145950134 IC50 > 30000 nM T81386 C7N3ZQ 145951035 IC50 > 10000 nM T81386 C9GBH4 145951220 IC50 > 30000 nM T81386 CML51F 145951743 IC50 > 10000 nM T81386 C0LA4N 145952248 IC50 > 30000 nM T81386 CN2OI4 145952973 IC50 > 30000 nM T81386 CEV70S 145953574 IC50 > 10000 nM T81386 CQR1T0 145957794 IC50 > 30000 nM T81386 CMJ5D9 145958016 IC50 > 10000 nM T81386 C42CGJ 145958217 IC50 = 220 nM T81386 CMH3Q4 145959803 IC50 = 15000 nM T81386 CT30CG 145960449 IC50 > 10000 nM T81386 CE9D6T 145960511 IC50 > 10000 nM T81386 C4M6SJ 145961986 IC50 > 10000 nM T81386 C36PIF 145963783 IC50 = 49 nM T81386 C6PQN3 145963970 IC50 = 6 nM T81386 CDF9U4 145964106 IC50 = 3 nM T81386 CZW3C9 145964690 IC50 = 1800 nM T81386 C87KPO 145964931 IC50 = 1 nM T81386 C93NOQ 145965274 IC50 = 2400 nM T81386 CN90GT 145965313 IC50 = 2 nM T81386 CI9KC4 145965423 IC50 = 2 nM T81386 C5V8PB 145965855 IC50 > 12500 nM T81386 CMZ63P 145965913 IC50 = 5 nM T81386 C9E4UT 145966185 IC50 = 14 nM T81386 CY19JM 145966214 IC50 > 12500 nM T81386 C3HZ8E 145966261 IC50 > 12500 nM T81386 CI21WV 145966399 IC50 = 10 nM T81386 C2Y6IZ 145966577 IC50 = 122 nM T81386 CT78XQ 145966753 IC50 = 3600 nM T81386 CBI23W 145967175 IC50 = 458 nM T81386 CSC1U2 145967972 IC50 = 5 nM T81386 CO7C1T 145969623 IC50 = 55 nM T81386 CNK98R 145970759 IC50 = 6 nM T81386 C9EO3S 145971368 IC50 = 378 nM T81386 CX9PG6 145972012 IC50 > 10000 nM T81386 C08DEY 145972145 IC50 = 529300 nM T81386 C92KLM 145972371 IC50 = 21 nM T81386 CSP5B8 145972813 IC50 = 8 nM T81386 CC8S9M 145972872 IC50 = 0.4 nM T81386 CJZ0B6 145972978 IC50 = 2400 nM T81386 CRHV10 145973338 IC50 = 9 nM T81386 CE0SV4 145973475 IC50 = 13 nM T81386 CBT27W 145973693 IC50 > 12500 nM T81386 CU9TI2 145973744 IC50 = 11 nM T81386 C2VK8B 145973776 IC50 = 10400 nM T81386 C1HKY6 145973930 IC50 = 2 nM T81386 C3MIA9 145973951 IC50 = 210 nM T81386 CSN17I 145974162 IC50 = 3 nM T81386 CX70JG 145974213 IC50 = 25 nM T81386 C02ZTX 145974441 IC50 = 4 nM T81386 C9M5YW 145974763 IC50 > 12500 nM T81386 CRJ23M 145974842 IC50 > 12500 nM T81386 CVA2M0 145975301 IC50 = 3500 nM T81386 C2FG9E 145975412 IC50 = 4 nM T81386 CPC83F 145975562 IC50 = 8 nM T81386 CQA87Y 145975607 IC50 = 1 nM T81386 C6SQL9 145975632 IC50 = 3 nM T81386 C5P3OR 145976229 IC50 = 12 nM T81386 CWG2J6 145976257 IC50 = 9 nM T81386 CP9M7T 145976565 IC50 = 33 nM T81386 C5W8GH 145976701 IC50 = 2 nM T81386 CBR9Q3 145976910 IC50 = 2 nM T81386 CNZT52 145977047 IC50 = 50 nM T81386 C3G5FY 145977120 IC50 = 12 nM T81386 C1NQ5F 145977131 IC50 = 135 nM T81386 CL58MT 145977187 IC50 > 12500 nM T81386 CBQ4S8 145977291 IC50 = 66 nM T81386 CCQS56 145977821 IC50 = 2 nM T81386 C9DCP3 145977923 IC50 > 12500 nM T81386 CQD9J5 145978289 IC50 = 17 nM T81386 C5UQ6Z 145978465 IC50 = 9 nM T81386 C0NWY6 145978593 IC50 = 1576 nM T81386 CX05ZN 145979845 IC50 = 890 nM T81386 CVES49 145982552 IC50 = 2000 nM T81386 CIDU48 145982789 IC50 > 10000 nM T81386 CPO43Z 145982872 IC50 > 10000 nM T81386 CORV50 145982985 IC50 = 700 nM T81386 C6YBK0 145983031 IC50 = 2000 nM T81386 CD3WR9 145983454 IC50 > 10000 nM T81386 CQXC48 145983553 IC50 > 10000 nM T81386 CJ4N1S 145983820 IC50 = 1500 nM T81386 C8GVD0 145984001 IC50 = 9000 nM T81386 CTJW32 145984202 IC50 = 420 nM T81386 C48YNJ 145985058 IC50 = 2100 nM T81386 C67EVF 145985214 IC50 = 1500 nM T81386 CKQ69G 145985465 IC50 = 700 nM T81386 C7CH9V 146014951 IC50 = 824 nM T81386 CRTP54 155301364 IC50 = 179 nM T81386 CUW29V 155301374 IC50 = 94.1 nM T81386 CC9WJ5 155301438 IC50 = 19.9 nM T81386 C4PIF7 155301446 IC50 = 10.8 nM T81386 CEAQ01 155510741 IC50 = 12 nM T81386 CJB1R5 155511461 IC50 > 20000 nM T81386 C2MD1Q 155513187 IC50 > 10000 nM T81386 CU9SG3 155515972 IC50 = 50 nM T81386 CE9N5W 155518278 IC50 = 34 nM T81386 CZ0WO7 155523990 IC50 = 16100 nM T81386 C5J8AS 155524785 IC50 > 10000 nM T81386 CHMV49 155525041 IC50 > 20000 nM T81386 C82MLZ 155526827 IC50 = 5 nM T81386 CQK49J 155527932 Ki > 5000 nM T81386 C42CYF 155529938 IC50 = 10 nM T81386 CH4R0A 155531793 IC50 = 42 nM T81386 C2M5JU 155532995 IC50 = 68 nM T81386 CN57JE 155534846 Ki > 5000 nM T81386 C9VK2Q 155537187 IC50 = 11 nM T81386 CQ8UA4 155538384 Ki > 5000 nM T81386 CVTD36 155539890 Ki > 5000 nM T81386 CAX3K4 155543060 Ki > 5000 nM T81386 CHD09S 155543566 IC50 = 5110 nM T81386 CVS1L8 155543641 IC50 = 9 nM T81386 CC6KQ2 155550557 IC50 = 15 nM T81386 C2VLU5 155551528 IC50 > 100000 nM T81386 CC5YK7 155552067 IC50 = 25 nM T81386 CWND70 155556435 IC50 = 12.7 nM T81386 CZ8D5Y 155556955 IC50 = 33 nM T81386 CQI5Z4 155558076 IC50 > 10000 nM T81386 CP7R2X 155558740 IC50 > 50000 nM T81386 CQ7BX0 155559110 Ki = 1000 nM T81386 C5G7IY 155563601 IC50 = 9 nM T81386 C1N8OX 155564817 IC50 > 100000 nM T81386 CN6SQ5 155567919 IC50 = 4 nM T81386 CEN7R1 155569345 IC50 = 6 nM T81386 D00HSJ 10275789 IC50 = 1.37 nM T81386 D00MXS 5281703 IC50 = 198 nM T81386 D01MNK 25125014 IC50 = 90 nM T81386 D01PEF 24801181 IC50 = 1200 nM T81386 D03YVL 5472558 IC50 > 20000 nM T81386 D04BNM 5894 Ki = 340 nM T81386 D04RBG 3536 IC50 = 540 nM T81386 D04UNQ 242623 IC50 = 15000 nM T81386 D04WFN 10202471 IC50 = 5100 nM T81386 D05SZH 135402864 IC50 = 1800 nM T81386 D07HPE 481747 IC50 > 20000 nM T81386 D07OCA 5330812 IC50 = 30 nM T81386 D08HFG 24809764 IC50 = 394 nM T81386 D08KSQ 11637090 IC50 = 26 nM T81386 D09OAH 73292 IC50 > 250000 nM T81386 D0A7FQ 11644425 Ki > 10000 nM T81386 D0B9YR 24801697 IC50 = 7 nM T81386 D0D0ZQ 24801185 IC50 = 5.6 nM T81386 D0D2FC 2794188 IC50 = 1400 nM T81386 D0D5HQ 5330797 IC50 = 4000 nM T81386 D0D5ZL 369401 IC50 = 810 nM T81386 D0E3FK 24801186 IC50 = 5300 nM T81386 D0H6CQ 23727982 IC50 = 5.6 nM T81386 D0L3FK 5289419 IC50 = 1500 nM T81386 D0LO5B 73602827 IC50 = 2831 nM T81386 D0N3LC 90643548 IC50 = 729 nM T81386 D0P2WA 6918386 IC50 = 2300 nM T81386 D0R5FH 438981 IC50 = 14100 nM T81386 D0RJ8J 76072859 IC50 = 749 nM T81386 D0S8VE 23727981 IC50 = 6 nM T81386 D0U1WL 24801699 IC50 = 18 nM T81386 D0VD8B 3004085 IC50 > 20000 nM T81386 D0Y0ES 3707 IC50 = 2400 nM T81386 D0Y5RO 4566 IC50 = 1070 nM T85799 D03MNN 11341869 IC50 > 1000 nM T85799 D04LVK 57379345 IC50 = 4720 nM T85799 D05SBO 46220502 IC50 = 2 nM T85799 D0B0AX 5328127 IC50 > 40000 nM T85799 D0W5HK 216239 IC50 > 3000 nM T85799 D00UZR 5330286 IC50 = 9 nM T85799 D03LWG 53235510 IC50 > 10000 nM T85799 D05ADP 160355 IC50 > 100000 nM T85799 D06WHY 16747683 IC50 = 450 nM T85799 D08MXP 44631912 IC50 = 2 nM T85799 D0CY1B 6420138 Ki = 1090 nM T85799 D0DX4J 67409219 IC50 < 100 nM T85799 D0LF1U 5287969 Ki = 40 nM T85799 D0S5RC 3025986 Ki = 925 nM T85799 D0Z1DH 10029385 IC50 = 1800 nM T85799 D00BPA 4592 IC50 > 100000 nM T85799 D0D3PX 46926350 IC50 = 127 nM T85799 D0Z0KD 5330258 IC50 < 20 nM T85799 C1BE5N 3799 IC50 < 10000 nM T85799 C28CSW 158883 IC50 = 1420 nM T85799 CV7W4J 176406 IC50 < 10000 nM T85799 C4MNG8 445840 IC50 = 42 nM T85799 CPRG75 447446 IC50 = 680 nM T85799 CNF1P5 447652 IC50 = 8900 nM T85799 CJA3D4 447958 Ki > 20000 nM T85799 CFDR89 447959 Ki = 210 nM T85799 CXS8U2 447960 Ki = 320 nM T85799 CB9F1O 447961 Ki = 53 nM T85799 C6A3LY 447962 Ki = 960 nM T85799 C1ZG2U 449087 IC50 > 10000 nM T85799 CFHO09 481744 IC50 = 6000 nM T85799 CNVT43 481745 IC50 = 6300 nM T85799 CM7NF4 481746 IC50 = 7000 nM T85799 CL15VX 481748 IC50 = 20000 nM T85799 C9Z7AU 3496894 IC50 = 100 nM T85799 CU5B1Z 4369491 IC50 = 3750 nM T85799 C7WXK1 4469813 IC50 = 6000 nM T85799 CAXZ94 4475481 IC50 = 800 nM T85799 C4DU1B 4475482 IC50 = 9000 nM T85799 CFEU51 4478473 IC50 = 100 nM T85799 C4MUT0 5289179 IC50 = 5053 nM T85799 CPT61U 5328112 IC50 > 50000 nM T85799 CDM98R 5328125 IC50 > 40000 nM T85799 CDY2O3 5328134 IC50 > 40000 nM T85799 CC1O0M 5328135 IC50 > 40000 nM T85799 C14LVT 5328137 IC50 > 40000 nM T85799 COT45A 5328149 IC50 > 40000 nM T85799 CTC68O 5329656 IC50 = 0.026 nM T85799 C8C3VG 5329674 IC50 = 1090 nM T85799 CM9V8E 5329715 IC50 = 6150 nM T85799 CW0Z9J 5329753 IC50 = 0.08 nM T85799 CBW30C 5330047 IC50 = 0.007 nM T85799 C5PL8M 5330199 IC50 = 620 nM T85799 CGI90W 5330278 IC50 = 5 nM T85799 CL5I2U 5330279 IC50 = 2 nM T85799 C4V5QX 5330356 IC50 < 20 nM T85799 CZ3LK2 5330387 IC50 > 10000 nM T85799 C5SY4O 5330420 IC50 > 10000 nM T85799 CUEZ35 5330437 IC50 > 10000 nM T85799 C5TGL0 5330583 IC50 = 2.3 nM T85799 CK4CO2 5330614 IC50 = 1081 nM T85799 CJI2G7 5330615 IC50 = 827 nM T85799 CH4IV5 5330616 IC50 = 838 nM T85799 C8LTE0 5330617 IC50 = 1973 nM T85799 CFD3I6 5330618 IC50 = 359 nM T85799 CE2X0C 5330619 IC50 = 1894 nM T85799 CE4I0K 5330620 IC50 = 786 nM T85799 C96AEG 5330621 IC50 = 464 nM T85799 CLXG43 5330622 IC50 = 2589 nM T85799 C16LYJ 5330623 IC50 = 1144 nM T85799 C3VZF8 5330624 IC50 = 810 nM T85799 C48LEV 5330625 IC50 = 1033 nM T85799 C5LVY9 5330627 IC50 = 1703 nM T85799 C6ROJ7 5330642 IC50 = 1553 nM T85799 C35TQR 5330890 IC50 = 74500 nM T85799 CPTX95 5330921 IC50 = 8300 nM T85799 CLJ1W5 5332196 IC50 = 0.75 ug.mL-1 T85799 C36XBW 5714753 IC50 > 20 ug.mL-1 T85799 CCRM28 6538898 IC50 = 4410 nM T85799 C0O8DH 6538899 IC50 = 25250 nM T85799 CW9S3K 6538900 IC50 = 2210 nM T85799 C5Y7MX 6538901 IC50 = 1870 nM T85799 CZH30S 6538902 IC50 = 1920 nM T85799 CK4HA1 6538931 IC50 = 33000 nM T85799 C3SVJ4 6538972 IC50 = 15000 nM T85799 C0N8IC 6538973 IC50 = 8000 nM T85799 C0R3HT 6538974 IC50 = 18000 nM T85799 C1JPE7 6538975 IC50 = 27000 nM T85799 C91GSM 6538976 IC50 = 8000 nM T85799 CD4ZY6 6538977 IC50 = 4000 nM T85799 C4KO2H 6538978 IC50 = 23000 nM T85799 C59NXD 6538979 IC50 = 2000 nM T85799 C18DCI 6538980 IC50 = 1000 nM T85799 CJMA92 6538981 IC50 = 50 nM T85799 CQU63M 6538982 IC50 = 500 nM T85799 CR62XM 6538983 IC50 = 800 nM T85799 C2HZQ7 6538984 IC50 = 5000 nM T85799 C9XQV0 6538985 IC50 = 2000 nM T85799 CEG54P 6538986 IC50 = 1000 nM T85799 C4APW5 6538987 IC50 = 1000 nM T85799 C48ERS 6538988 IC50 = 1000 nM T85799 CFA5Z0 6538989 IC50 = 2000 nM T85799 CA68PN 6538990 IC50 = 19000 nM T85799 C8YH9W 6538991 IC50 = 2000 nM T85799 C6V0LQ 6538992 IC50 = 1000 nM T85799 C76LEK 6538993 IC50 = 2000 nM T85799 CBO5S8 6538994 IC50 = 2000 nM T85799 C4D0WX 6538995 IC50 = 700 nM T85799 CS6DQ2 6538996 IC50 = 2000 nM T85799 CH04KA 6538997 IC50 = 600 nM T85799 CRH42M 6538998 IC50 = 100 nM T85799 CZ2PE0 6538999 IC50 = 200 nM T85799 CXW9Y6 6539000 IC50 = 300 nM T85799 C8CSQ3 6539001 IC50 = 1000 nM T85799 CU8PL7 6539002 IC50 = 200 nM T85799 CH70WZ 6539003 IC50 = 800 nM T85799 CXF78K 6539004 IC50 = 300 nM T85799 C3E2VM 6539005 IC50 = 100 nM T85799 CK7O9B 6539006 IC50 = 10 nM T85799 C6R2TO 6539007 IC50 = 40000 nM T85799 CZ7F0B 6539008 IC50 > 10000 nM T85799 CWP7M9 6539009 IC50 = 3600 nM T85799 CT9XA5 6539010 IC50 = 150 nM T85799 C1MGU7 6539011 IC50 = 2500 nM T85799 C6MDN7 6539012 IC50 = 41000 nM T85799 C47VIS 6539013 IC50 = 57000 nM T85799 CS8VA4 6539014 IC50 = 25000 nM T85799 C2Z8SX 6539015 IC50 = 4000 nM T85799 C04YNQ 6539016 IC50 = 2000 nM T85799 C5WK8I 6539017 IC50 = 2700 nM T85799 CS6VL5 6539018 IC50 = 8000 nM T85799 C0L5BW 6539026 IC50 = 3100 nM T85799 CW9MN4 6539027 IC50 = 260 nM T85799 C6MRY3 6539278 Ki > 20000 nM T85799 CXQ92S 6539279 Ki > 20000 nM T85799 CEL82X 6539280 Ki = 2600 nM T85799 CU2N3Q 6539281 Ki > 20000 nM T85799 CN1AU7 6539282 Ki = 9400 nM T85799 C6IB7U 6539283 Ki > 20000 nM T85799 CC62GN 6539284 Ki = 1200 nM T85799 C0J8QA 6539285 Ki = 900 nM T85799 CR8KA0 6539286 Ki > 20000 nM T85799 C9P5OX 6539287 Ki > 20000 nM T85799 C3KM1T 6539288 Ki > 20000 nM T85799 C8OC9M 6539289 Ki = 370 nM T85799 C7IWS5 6539290 Ki > 20000 nM T85799 CM35CV 6539291 Ki = 320 nM T85799 CT7MP9 6539292 Ki = 320 nM T85799 C1CRW6 6539293 Ki > 20000 nM T85799 C3HQ1G 6539294 Ki > 20000 nM T85799 CQ9U3J 6539295 Ki = 5300 nM T85799 COL0X2 6539296 Ki = 1600 nM T85799 CKV60H 6539297 Ki = 7100 nM T85799 CBC56F 6539298 Ki > 20000 nM T85799 C0LMW1 6539299 Ki > 20000 nM T85799 C51VJH 6539300 Ki = 10640 nM T85799 C0K1VF 6539301 Ki = 480 nM T85799 C95ETX 6539302 Ki = 270 nM T85799 CY03LO 6539303 Ki = 1000 nM T85799 CO8NR2 6539304 Ki = 900 nM T85799 CN76AU 6539305 Ki = 4170 nM T85799 C6UZF0 6539306 Ki = 960 nM T85799 C84MNG 6539307 Ki = 180 nM T85799 C38NYA 6539308 Ki = 260 nM T85799 C08SLD 6539309 Ki = 180 nM T85799 C6VB9U 6539310 Ki = 220 nM T85799 CB6N1Y 6539311 Ki = 300 nM T85799 CKJW72 6539312 Ki = 900 nM T85799 CQV1J5 6539313 Ki = 420 nM T85799 C1M4LA 6539314 Ki = 120 nM T85799 CO4QV9 6539315 Ki = 1910 nM T85799 C96XMO 6539316 Ki = 1600 nM T85799 CM2N8O 6539359 IC50 = 12 nM T85799 CUK02R 6539362 IC50 = 25 nM T85799 CZY97M 6539363 IC50 = 8 nM T85799 C9X8DW 6539364 Ki = 1990 nM T85799 CM9FT4 6539365 Ki = 310 nM T85799 C9Y3KC 6539366 Ki = 1990 nM T85799 C6Z0WU 6539368 Ki = 790 nM T85799 CY1W7D 6539369 Ki = 10 nM T85799 C8RND3 6539371 Ki = 310 nM T85799 CB69DA 6539372 Ki = 1990 nM T85799 CL18KE 6539373 Ki = 10 nM T85799 C74TAS 6539375 Ki = 190 nM T85799 C2GFT6 6539376 Ki = 250 nM T85799 C7SHN5 6539377 Ki = 60 nM T85799 CQM14U 6539378 Ki = 1990 nM T85799 CTBE09 6539379 Ki = 1580 nM T85799 CN2XV5 6539381 Ki > 19950 nM T85799 CQ84MY 6539384 Ki > 19950 nM T85799 C5Z4AQ 6539385 Ki > 19950 nM T85799 CZQ56A 6539386 Ki = 150 nM T85799 CA5YC3 6539387 Ki = 100 nM T85799 C6A0FQ 6539388 Ki > 19950 nM T85799 CX0T4J 6539389 Ki > 19950 nM T85799 CYC62P 6539392 Ki = 1580 nM T85799 C9NC7H 6539393 Ki = 30 nM T85799 CU85HS 6539395 Ki = 390 nM T85799 CQ51SX 6539396 Ki = 70 nM T85799 CVU8N0 6918710 IC50 = 80 nM T85799 C0QF4S 9800769 IC50 = 11 nM T85799 CQX25A 9858131 IC50 = 480 nM T85799 CRC65X 9863786 IC50 > 25000 nM T85799 CM5Z8X 9869943 IC50 > 100000 nM T85799 C3HG2L 9924275 IC50 = 170 nM T85799 C57URF 9951265 IC50 = 3700 nM T85799 CHFO23 9994136 IC50 = 6700 nM T85799 CVE1W8 10024433 Ki = 929 nM T85799 CZP6U0 10110571 IC50 = 1800 nM T85799 C50QLR 10110675 IC50 = 1750 nM T85799 CXBW34 10114553 IC50 = 2200 nM T85799 CO6E1A 10125856 IC50 = 160 nM T85799 C0H9JX 10125875 IC50 = 1000 nM T85799 CTXW95 10126509 IC50 = 12 nM T85799 CGT4F0 10134861 IC50 = 3000 nM T85799 CL2F5J 10135889 IC50 = 2000 nM T85799 CPT91S 10138993 IC50 = 750 nM T85799 CDTB71 10151417 IC50 = 800 nM T85799 C08VYL 10158127 IC50 = 1050 nM T85799 C79SUC 10158868 IC50 = 1300 nM T85799 C68GUB 10159114 IC50 = 3000 nM T85799 C8YZL0 10171618 IC50 = 2000 nM T85799 CQG5R4 10173796 IC50 = 6 nM T85799 CLE8V6 10182312 IC50 = 1800 nM T85799 CY7W5M 10192938 IC50 = 200 nM T85799 CYG69U 10193464 IC50 = 400 nM T85799 CHP56L 10193482 IC50 = 3200 nM T85799 CW2Y7N 10200092 IC50 = 2200 nM T85799 CIGT47 10202305 IC50 = 1600 nM T85799 CVRO56 10204194 IC50 = 2000 nM T85799 C7MVB8 10214675 IC50 = 800 nM T85799 C51UXK 10215135 IC50 = 500 nM T85799 COWF65 10215271 IC50 = 0.3 nM T85799 C5V6PK 10216157 IC50 = 50 nM T85799 CE2G4B 10216381 IC50 = 25 nM T85799 CHM97B 10221628 IC50 = 4000 nM T85799 CLW0H7 10223662 IC50 = 1300 nM T85799 C6NV7Q 10236923 IC50 = 250 nM T85799 CTS43G 10238877 IC50 = 26 nM T85799 CH48JA 10239038 IC50 = 38 nM T85799 C1KX3P 10248401 Ki = 2170 nM T85799 CG65JV 10275574 IC50 = 1400 nM T85799 C8GJ9A 10286242 IC50 = 1000 nM T85799 CDG1X4 10286382 IC50 > 40000 nM T85799 C42MKP 10286399 IC50 = 1600 nM T85799 C2O4LF 10286648 IC50 = 250 nM T85799 C9BH4P 10292184 IC50 = 6 nM T85799 C85MHR 10297090 IC50 > 1000 nM T85799 C6PL7N 10297469 IC50 = 1330 nM T85799 CZS4V6 10308171 IC50 = 1300 nM T85799 C9MVA5 10308281 IC50 = 2000 nM T85799 CKA8B0 10308522 IC50 = 4 nM T85799 COD9W2 10308706 IC50 = 790 nM T85799 C6S9AO 10310395 IC50 = 45 nM T85799 C9J3RM 10320107 Ki = 22 nM T85799 CMY9D2 10340715 Ki = 196 nM T85799 CC3L8Z 10430000 Ki = 943 nM T85799 CT0O5K 10634145 IC50 > 50 ug.mL-1 T85799 CK2ZP3 10805953 IC50 > 50 ug.mL-1 T85799 C94QUD 11163861 Ki = 10 nM T85799 C30PKR 11248978 IC50 = 1700 nM T85799 CSXY78 11294864 IC50 = 4800 nM T85799 CPU9I3 11316975 IC50 = 1500 nM T85799 CQ8I4H 11328863 IC50 = 3300 nM T85799 C7HMO6 11526786 IC50 > 50000 nM T85799 CIWA03 11632150 Ki = 666 nM T85799 CEV5X2 11646645 Ki = 38 nM T85799 C2CVI7 11647020 Ki > 10000 nM T85799 C93KHF 11718021 Ki = 955 nM T85799 C28TNJ 11722322 IC50 = 5600 nM T85799 CJSV21 11744184 Ki > 10000 nM T85799 C2Z8DQ 14624081 IC50 = 400 nM T85799 C7BS2R 16037674 IC50 = 34 nM T85799 CB2H4D 16037675 IC50 = 9.2 nM T85799 C9TU1O 16046126 IC50 = 6.4 nM T85799 CVS0T5 17754396 IC50 > 10000 nM T85799 CCF2B3 17933136 IC50 > 8600 nM T85799 C9RUO2 22273524 IC50 = 5600 nM T85799 CQHK69 23646624 IC50 = 31 nM T85799 CH1B7R 23646625 IC50 = 600 nM T85799 C8TIN5 23646628 IC50 = 1000 nM T85799 C9ZS1H 23646629 IC50 = 29 nM T85799 C50QUN 23646630 IC50 = 340 nM T85799 CS3UY4 23646631 IC50 = 1400 nM T85799 CR7JY4 23646632 IC50 = 2000 nM T85799 CIM15C 23646633 IC50 = 2100 nM T85799 CJUK39 24770517 IC50 > 10000 nM T85799 C9PA0M 24807809 IC50 > 50000 nM T85799 CZ48LS 24825971 IC50 = 1500 nM T85799 C13QYB 24884503 IC50 > 2000 nM T85799 CYDU89 24884773 IC50 = 530 nM T85799 CE2MR9 24884776 IC50 = 140 nM T85799 CB0V4I 24963033 IC50 = 200 nM T85799 CD5HQ0 24969301 IC50 > 10000 nM T85799 CMSW41 44361566 IC50 = 6700 nM T85799 C9M3GP 44361567 IC50 = 3000 nM T85799 CSBC59 44396134 IC50 = 18000 nM T85799 C54JRW 44399701 IC50 = 2 nM T85799 CUY8A3 44401410 IC50 = 260 nM T85799 C8L5ZH 44401437 IC50 = 29 nM T85799 CIB5V1 44401506 IC50 = 260 nM T85799 C5C3BG 44401556 IC50 = 57 nM T85799 C5HZF2 44413509 IC50 = 4.2 nM T85799 C3D4FG 44413527 IC50 = 13 nM T85799 CFED20 44415457 IC50 = 47 nM T85799 C2OFP6 44416439 IC50 = 6 nM T85799 C8JT0Q 44416469 IC50 = 13 nM T85799 CEIX01 44416574 IC50 = 160 nM T85799 C5NO1J 44416598 IC50 = 3.6 nM T85799 CO42UK 44416618 IC50 = 11 nM T85799 CZ3IU7 44416620 IC50 = 29 nM T85799 C8AP5N 44416899 IC50 > 10000 nM T85799 C9UC3V 44417819 IC50 = 110 nM T85799 C47YDK 44417820 IC50 = 350 nM T85799 CB9RV2 44447912 IC50 = 710 nM T85799 C4MQJ7 44447913 IC50 = 890 nM T85799 C2N6CE 44447930 IC50 = 210 nM T85799 CJC85A 44565069 IC50 = 6600 nM T85799 C5TE0I 44575454 IC50 = 32 ug.mL-1 T85799 C1ARI6 44575455 IC50 = 12 ug.mL-1 T85799 C5I3HT 44580807 IC50 = 16 nM T85799 CMH2A3 44580824 IC50 = 160 nM T85799 CTP7I4 44580861 IC50 = 8 nM T85799 C4JKW3 44581167 IC50 = 12 nM T85799 C2ZVF5 44589014 IC50 > 9000 nM T85799 C7ND9J 44589042 IC50 = 1500 nM T85799 CU47KI 44589090 IC50 = 490 nM T85799 CTY03Z 44589091 IC50 = 210 nM T85799 C4R5DC 44590971 IC50 > 20 ug.mL-1 T85799 CTMD40 44590972 IC50 = 4.4 ug.mL-1 T85799 C36LEO 44590973 IC50 = 3.2 ug.mL-1 T85799 C1PY6R 44590974 IC50 = 0.88 ug.mL-1 T85799 CMH56U 44590975 IC50 = 0.55 ug.mL-1 T85799 CF0LH6 44590976 IC50 = 0.24 ug.mL-1 T85799 C0KTA3 44590977 IC50 = 0.47 ug.mL-1 T85799 CZ5OJ9 44591009 IC50 = 0.39 ug.mL-1 T85799 CC80SY 44591092 IC50 = 0.9 ug.mL-1 T85799 CB8JF4 44591093 IC50 = 0.5 ug.mL-1 T85799 C0QJE3 44591094 IC50 = 0.88 ug.mL-1 T85799 CG5S0Z 44591095 IC50 = 0.52 ug.mL-1 T85799 C42IQG 44591096 IC50 = 0.59 ug.mL-1 T85799 CX5G9N 44591097 IC50 = 0.25 ug.mL-1 T85799 C28VWN 44591131 IC50 = 0.056 ug.mL-1 T85799 CH7VJ6 44591132 IC50 = 0.17 ug.mL-1 T85799 CH4Y1M 44591133 IC50 = 0.35 ug.mL-1 T85799 C3JVS0 44591386 IC50 = 1.9 ug.mL-1 T85799 CEK87I 44591387 IC50 = 0.05 ug.mL-1 T85799 CAY1Z9 44591388 IC50 = 0.12 ug.mL-1 T85799 CYR7B1 44591389 IC50 > 20 ug.mL-1 T85799 CD9G1Q 44591421 IC50 = 16 ug.mL-1 T85799 C57SZQ 44591422 IC50 > 20 ug.mL-1 T85799 C8NL6S 44591423 IC50 > 20 ug.mL-1 T85799 CQ5R0Z 44591424 IC50 > 20 ug.mL-1 T85799 C3FVR5 44591425 IC50 = 2.8 ug.mL-1 T85799 CC2WT4 46232590 IC50 = 9000 nM T85799 CGO1J5 46830766 Ki = 840 nM T85799 CF7HK2 46830767 Ki = 807 nM T85799 C2HJ1X 46830768 Ki = 1248 nM T85799 C7H4YM 46865419 IC50 > 10000 nM T85799 C2B5XF 49765254 IC50 = 324 nM T85799 CT0G4R 49800100 IC50 = 223 nM T85799 CWB4T2 49840036 IC50 = 451 nM T85799 C1MAO5 49840175 IC50 = 134 nM T85799 CJZ5A0 49840306 IC50 = 468 nM T85799 CCL3R5 49867929 IC50 = 33000 nM T85799 CG85OC 52940761 IC50 > 2100 nM T85799 C8BOP9 52942870 IC50 = 260 nM T85799 C0UC1B 52943026 IC50 = 150 nM T85799 CY8V0Q 52949108 IC50 = 810 nM T85799 C6BPR2 58985201 IC50 > 50000 nM T85799 CFD0Q4 60202647 IC50 = 23 nM T85799 CR2T5Q 66934034 Ki < 100 nM T85799 CJY4P6 68212724 IC50 = 199 nM T85799 CBE67N 71731769 IC50 > 10000 nM T85799 CYG95S 72707651 IC50 = 42 nM T85799 CNP0V5 72707724 IC50 = 40 nM T85799 CU4A5Q 72707728 IC50 = 40 nM T85799 CZAM98 72707790 IC50 = 39 nM T85799 CP13FK 72707853 IC50 = 35 nM T85799 C9MPZ1 77107163 IC50 = 23 nM T85799 C7VA5U 78161839 IC50 > 10000 nM T85799 C8W9KV 91844733 IC50 = 49000 nM T85799 C8UL7Y 122657565 IC50 = 7.4 nM T85799 CHT7A6 122657605 IC50 = 0.8 nM T85799 C6J5BQ 122657629 IC50 = 0.6 nM T85799 C0NPF8 122657632 IC50 = 18 nM T85799 CSW6L2 122667245 IC50 = 35.9 nM T85799 C63VIC 122667249 IC50 = 1.6 nM T85799 CEG56K 122667252 IC50 = 2.4 nM T85799 C3J9UR 122667253 IC50 = 13.8 nM T85799 C1SDO8 122667293 IC50 = 2.9 nM T85799 CLHF95 122667296 IC50 = 2.1 nM T85799 CKA47Z 122667297 IC50 = 5156 nM T85799 C5R4PU 122667312 IC50 = 5.2 nM T85799 CG8ZM5 122667313 IC50 = 12.1 nM T85799 CAQP38 122667319 IC50 = 1.5 nM T85799 CA3KV2 122667321 IC50 = 283.4 nM T85799 CAJH71 122667328 IC50 = 5.6 nM T85799 CSY3M0 122667329 IC50 = 2.2 nM T85799 CJU5O4 122667350 IC50 = 3.7 nM T85799 C09GPH 122667359 IC50 = 2.9 nM T85799 CW95MK 122667361 IC50 = 1.6 nM T85799 CZT1C4 122667385 IC50 = 3.1 nM T85799 CR5MA6 122667387 IC50 = 8.8 nM T85799 C1SP3H 127030849 IC50 > 2000 nM T85799 CVB7D2 129102568 IC50 = 16 nM T85799 C9BOH1 129102571 IC50 = 20 nM T85799 C4T9DH 129102574 IC50 = 5.7 nM T85799 CJ25TP 129102576 IC50 = 25 nM T85799 C8U9SE 129102577 IC50 = 9.7 nM T85799 CBOS93 129102582 IC50 = 49.7 nM T85799 C32QTR 129102589 IC50 = 0.6 nM T85799 C1GJQ3 129102591 IC50 = 14 nM T85799 CZAB64 129102594 IC50 = 27 nM T85799 CXO0V7 129102595 IC50 = 39 nM T85799 C6Y7VA 129102598 IC50 = 5.7 nM T85799 C72GIC 129102599 IC50 = 15.8 nM T85799 C8EIU5 129102600 IC50 = 10 nM T85799 C06GCP 129102608 IC50 = 17.6 nM T85799 CL0VI3 129102610 IC50 = 147.3 nM T85799 C3AM4Y 129102611 IC50 = 1 nM T85799 CSTL63 129102640 IC50 = 6.8 nM T85799 C5M7PZ 129102643 IC50 = 1.72 nM T85799 C1H5GP 129102646 IC50 = 18.9 nM T85799 CW41KL 134135943 IC50 = 13 nM T85799 CJ3M5I 134137436 Ki > 1000 nM T85799 CFM28H 134144635 IC50 = 25 nM T85799 C5PE1B 134153020 IC50 = 32 nM T85799 C48DGU 134156416 IC50 = 19 nM T85799 CLSE63 135398512 IC50 > 10000 nM T85799 CS4OW8 135400873 Ki > 2000 nM T85799 COYA04 135402863 IC50 = 10000 nM T85799 CM4J6A 135444580 IC50 = 303 nM T85799 CV2RZ4 135464244 IC50 = 12500 nM T85799 CFAD48 135611170 Ki > 2000 nM T85799 C2EL8Y 135800267 IC50 < 10000 nM T85799 C3DNL6 137349544 IC50 = 42000 nM T85799 CU9O3A 137628639 IC50 = 22.5 nM T85799 C25ERN 137631967 IC50 > 1000 nM T85799 C8GQD5 137636872 IC50 = 441 nM T85799 C06JRX 137637094 IC50 > 1000 nM T85799 C1DK0P 137651391 IC50 > 1000 nM T85799 CV5H3Z 137657932 IC50 > 1000 nM T85799 C1LK7M 145975810 IC50 = 18.3 nM T85799 CR2GW6 145994117 IC50 > 5000 nM T85799 C42TMN 155523743 IC50 = 0.2 nM T85799 CM0U3I 155534552 IC50 = 417 nM T85799 CWM03V 155563050 IC50 > 20000 nM T85799 CAO81F 155563443 IC50 = 23000 nM T85799 CLXN40 155565350 IC50 = 21 nM T85799 D01MNK 25125014 IC50 = 20000 nM T85799 D02DLC 6539361 Ki = 60 nM T85799 D04TLB 135408762 IC50 = 230 nM T85799 D07HPE 481747 IC50 = 6000 nM T85799 D08RZB 11153014 IC50 > 25000 nM T85799 D09OAH 73292 IC50 = 350 nM T85799 D0D6MH 11617559 IC50 > 19000 nM T85799 D0D9PD 11656591 IC50 > 5000 nM T85799 D0G2CT 3708 IC50 = 200 nM T85799 D0GN5Z 5281295 IC50 = 2820 nM T85799 D0H3EV 5005498 IC50 > 10000 nM T85799 D0L3FK 5289419 IC50 = 200 nM T85799 D0O0VP 6539367 Ki = 190 nM T85799 D0P6JS 11675054 IC50 = 50 nM T85799 D0R1FT 4564 Ki > 100 nM T85799 D0T4SJ 10356352 IC50 = 1420 nM T85799 D0T8NU 16757525 IC50 > 4000 nM T85799 D0U0GE 447956 Ki = 16000 nM T85799 D0Y5RO 4566 IC50 = 1600 nM T85799 D0YZ7H 9797370 IC50 > 100000 nM T33367 CA98PG 258671 IC50 > 100000 nM T33367 CKS40E 258877 IC50 > 100000 nM T33367 CXO40G 728709 IC50 > 100000 nM T33367 CU6QR3 762797 IC50 > 100000 nM T33367 C72HMQ 831831 IC50 > 100000 nM T33367 C97RUC 851835 IC50 > 100000 nM T33367 C4XFW3 888738 IC50 > 100000 nM T33367 CNV74B 2195029 IC50 = 36000 nM T33367 CWY7L8 2802659 IC50 = 16000 nM T33367 C93BJK 2802661 IC50 > 100000 nM T33367 C9J5XH 2802665 IC50 = 8200 nM T33367 CLJ91H 2804574 IC50 = 36000 nM T33367 CQB72H 2818038 IC50 = 85000 nM T33367 CIA56C 3303561 IC50 = 63000 nM T33367 CV60AY 4086855 IC50 > 100000 nM T33367 C9K1CH 4207719 IC50 = 67000 nM T33367 CMVZ19 4803262 IC50 = 62000 nM T33367 C95ODG 11151251 IC50 > 100000 nM T33367 C3BV8R 13236629 IC50 > 100000 nM T33367 C0Y6DF 16189290 IC50 > 100000 nM T33367 CCX03M 17185449 IC50 > 100000 nM T33367 CZ4A6E 19057623 IC50 > 100000 nM T33367 CO6XB4 23604723 IC50 = 34000 nM T33367 CK6OZ0 24020563 IC50 = 32000 nM T33367 CA67WE 44755432 IC50 > 100000 nM T33367 C7OHZ1 52592583 IC50 = 39000 nM T33367 CC1E6W 86020022 IC50 > 100000 nM T33367 C4R5WH 86057524 IC50 > 100000 nM T33367 C5RHK6 108870201 IC50 = 28000 nM T33367 CB07HE 134108783 IC50 > 100000 nM T33367 C4DHP3 145982548 IC50 > 100000 nM T33367 C8XY4M 145982595 IC50 > 100000 nM T33367 CEFU35 145982611 IC50 = 43000 nM T33367 CQ65JM 145982672 IC50 > 100000 nM T33367 C2T7GO 145982723 IC50 = 64000 nM T33367 CCE7W5 145982759 IC50 = 21000 nM T33367 C15NKZ 145982777 IC50 > 100000 nM T33367 CS10FG 145982812 IC50 > 100000 nM T33367 C7GBW8 145982962 IC50 > 100000 nM T33367 CCXF72 145983066 IC50 = 36000 nM T33367 CE79BN 145983088 IC50 = 16000 nM T33367 C2L5OA 145983117 IC50 > 100000 nM T33367 CZ7WU8 145983149 IC50 > 100000 nM T33367 CG8KZ5 145983161 IC50 > 100000 nM T33367 C59OBK 145983227 IC50 > 100000 nM T33367 CXML60 145983274 IC50 = 25000 nM T33367 C96ATW 145983305 IC50 > 100000 nM T33367 C6ZVK0 145983309 IC50 > 100000 nM T33367 C2CG7Y 145983378 IC50 = 22000 nM T33367 CJ96OE 145983470 IC50 > 100000 nM T33367 CU1RQ4 145983473 IC50 = 39000 nM T33367 CB3S6Z 145983503 IC50 > 100000 nM T33367 CL74BO 145983521 IC50 > 100000 nM T33367 CD6IQ3 145983599 IC50 = 46000 nM T33367 CXV0T2 145983952 IC50 > 100000 nM T33367 C27AXM 145983955 IC50 > 100000 nM T33367 C2Z3EM 145984007 IC50 > 100000 nM T33367 CY5A7W 145984017 IC50 = 56000 nM T33367 C94FGA 145984079 IC50 > 100000 nM T33367 C0BY1H 145984097 IC50 = 52000 nM T33367 CNCU35 145984182 IC50 = 16000 nM T33367 CEC8T1 145984186 IC50 > 100000 nM T33367 CCQ1O3 145984238 IC50 > 100000 nM T33367 C9BIX3 145984279 IC50 > 100000 nM T33367 C9SLU7 145984283 IC50 > 100000 nM T33367 CI76FA 145984328 IC50 > 100000 nM T33367 CZ1JH0 145984468 IC50 = 41000 nM T33367 C8CQ9W 145984500 IC50 > 100000 nM T33367 CF6C0K 145984528 IC50 = 14000 nM T33367 CGB20S 145984549 IC50 > 100000 nM T33367 CQB7P2 145984574 IC50 > 100000 nM T33367 CL79BQ 145984794 IC50 > 100000 nM T33367 CED0V7 145984873 IC50 > 100000 nM T33367 CA60ZM 145985000 IC50 = 76000 nM T33367 CK7U8L 145985007 IC50 > 100000 nM T33367 C8C7EQ 145985087 IC50 > 100000 nM T33367 C2GX6Y 145985199 IC50 > 100000 nM T33367 C3NV1X 145985232 IC50 > 100000 nM T33367 CCA60N 145985239 IC50 > 100000 nM T33367 C7GH4B 145985328 IC50 > 100000 nM T33367 CHX97L 145985440 IC50 > 100000 nM T33367 CK4PL1 145985450 IC50 > 100000 nM T33367 CM8DT7 145985526 IC50 > 100000 nM T33367 CYPI79 145985566 IC50 > 100000 nM T33367 CJ1A6S 145985666 IC50 > 100000 nM T33367 C07VLB 145985670 IC50 > 100000 nM T33367 CY3Z5A 145985767 IC50 > 100000 nM T33367 C7L8VM 145985914 IC50 > 100000 nM T33367 CLCI62 145985930 IC50 > 100000 nM T33367 CC7S2J 145985996 IC50 > 100000 nM T33367 C0Q1YX 145986034 IC50 > 100000 nM T33367 C0X1GM 145986112 IC50 > 100000 nM T33367 CKLY90 145986283 IC50 > 100000 nM T99665 D03KEK 3765 EC50 = 38904.51 nM T99665 D0Q5IN 727 IC50 = 91 nM T99665 D0Y7ZD 137 IC50 = 12900 nM T99665 D01RBR 130021 IC50 = 62000 nM T99665 D0C9XA 119 EC50 = 269.15 nM T99665 D0Z8IJ 4266 EC50 = 691.83 nM T99665 CU3EJ0 96215 EC50 = 4570.88 nM T99665 CXSD61 155246 EC50 = 3800 nM T99665 CNV85P 928193 EC50 = 65000 nM T99665 C58SGV 1502041 EC50 = 20000 nM T99665 CW6QE8 1502042 EC50 = 9000 nM T99665 CDK8I7 1502043 EC50 = 59000 nM T99665 CRN61G 1502044 EC50 = 40000 nM T99665 C1A0UL 1502074 EC50 = 8317.64 nM T99665 CQ2C8G 2733883 EC50 = 19100 nM T99665 C5RM2I 5310987 EC50 = 400 nM T99665 CL30TV 6443915 EC50 = 2430 nM T99665 CVJ5L9 6971281 EC50 = 44800 nM T99665 CK86RB 10219459 IC50 = 5500 nM T99665 CZ0B5I 10240915 EC50 = 1584.89 nM T99665 CK0SV2 11286468 IC50 = 6600 nM T99665 CT5LD3 11819163 EC50 = 1230.27 nM T99665 CV41XS 12309465 IC50 = 800 nM T99665 CGA06Q 22019116 EC50 > 1000000 nM T99665 C62OLQ 22099243 IC50 = 300000 nM T99665 CIE27X 28881819 EC50 = 40000 nM T99665 C1RFE4 28881824 IC50 = 890000 nM T99665 C8UTR2 67642717 EC50 = 2754.23 nM T99665 CE4RJ7 68419998 EC50 > 1000000 nM T99665 C81NCF 71561429 EC50 > 500000 nM T99665 C12SFB 71561435 EC50 > 500000 nM T99665 C6EZ3X 71561439 EC50 > 500000 nM T99665 CC7D8K 71561443 EC50 > 500000 nM T99665 C0ZH1E 71561568 EC50 > 500000 nM T99665 C1VI4L 71582755 EC50 = 3090.3 nM T99665 C2T6DL 71717372 EC50 > 500000 nM T99665 C60HIG 71719189 EC50 > 500000 nM T99665 CS5WO3 71746803 IC50 = 12900 nM T99665 CH60SC 71746804 IC50 = 81500 nM T99665 C3XPG0 71746805 IC50 = 153000 nM T99665 C6QB1L 71746977 IC50 = 115300 nM T99665 CE23HJ 71746978 IC50 = 9600 nM T99665 C26OQL 71746979 IC50 = 408300 nM T99665 CIM9S4 71746980 IC50 = 570000 nM T99665 C6AI4G 118710364 EC50 > 1000000 nM T99665 CDR85F 118710366 EC50 > 1000000 nM T99665 CI7S8H 155516242 EC50 = 1584.89 nM T99665 C4U8QT 155524561 IC50 = 300000 nM T99665 CJ4OV6 155530359 EC50 = 1200 nM T99665 CEP10B 155553507 EC50 = 5370.32 nM T99665 CGF4Y0 155556567 EC50 = 3700 nM T99665 CL2Q6G 155567178 IC50 = 100000 nM T99665 D02ANG 5216267 EC50 = 6456.54 nM T99665 D0B5HD 3352 IC50 > 10000 nM T99665 D0C7PZ 22359367 EC50 = 22000 nM T99665 D0N4EZ 193060 EC50 = 4600 nM T99665 D0O4IM 928194 IC50 = 16000 nM T99665 D0O9UH 6603697 EC50 = 74000 nM T99665 D0U4HM 5521 IC50 = 2220 nM T99665 D0WZ9T 5310934 IC50 = 5400 nM T16188 D0E3TC 44259 IC50 = 4.2 nM T16188 C3VRO9 44557921 IC50 > 10000 nM T16188 CV63UL 67240318 IC50 > 10000 nM T16188 C2MD1Q 155513187 IC50 > 10000 nM T12808 D06GDY 43815 IC50 = 220000 nM T12808 D0AZ3C 5291 IC50 > 100000 nM T12808 D0E6XR 3062316 IC50 > 50000 nM T12808 D0EG1I 9926791 IC50 > 10000 nM T12808 D0J9ZR 4477 IC50 > 100000 nM T12808 D02RJY 11442891 IC50 > 10000 nM T12808 D03LWG 53235510 IC50 > 10000 nM T12808 D06IPZ 49800096 IC50 = 59000 nM T12808 D07EHV 44814409 IC50 > 10000 nM T12808 D09DHT 27924 Ki = 2.5 nM T12808 D0E3TC 44259 IC50 = 0.37 nM T12808 D0E6AH 5280757 Ki = 0.48 nM T12808 D0HS5V 11234052 IC50 > 25000 nM T12808 D0I6VU 176167 IC50 = 800 nM T12808 D0L4FS 5280961 IC50 > 100000 nM T12808 D0LF1U 5287969 IC50 = 2800 nM T12808 D0P1CV 46191454 IC50 > 10000 nM T12808 D0R9IU 44462758 IC50 = 90 nM T12808 D0S5RC 3025986 IC50 > 40000 nM T12808 D0U3EP 445154 EC50 = 5780000 nM T12808 D0W3LI 153999 IC50 = 360 nM T12808 D03BNU 59604787 IC50 > 10000 nM T12808 D0LF0O 135441202 IC50 = 11000 nM T12808 D0WS1V 448991 IC50 > 100000 nM T12808 D0A3MV 448014 IC50 > 100000000 nM T12808 D01EFO 9864718 IC50 = 72000 nM T12808 D04FHB 6918852 Ki > 5000 nM T12808 D08OTG 5281800 IC50 = 9300 nM T12808 D0A9KI 9863367 IC50 = 83 nM T12808 D0B3CT 9928668 IC50 = 40000 nM T12808 D0Q7HO 4705 IC50 > 100000 nM T12808 D0R5ZR 127757 IC50 = 22 nM T12808 D0T3ME 156422 IC50 > 30000 nM T12808 C8OI7N 2290 IC50 = 30 nM T12808 C95GCZ 3568 IC50 = 43000 nM T12808 C8NW5J 3815 IC50 = 2450 nM T12808 C79ZQW 73110 IC50 > 100000 nM T12808 C4UF9R 121295 IC50 = 11000 nM T12808 C7SD9A 129831 IC50 = 3590000 nM T12808 C1PMA7 130351 IC50 = 54000 nM T12808 CG2P1X 159320 Ki = 0.5 nM T12808 C8PU1O 188534 Ki = 5.8 nM T12808 CMN15U 192686 IC50 = 37000 nM T12808 C05NEZ 271592 Ki = 7800 nM T12808 C0T8ME 282272 Ki = 26600 nM T12808 C2IX3S 314520 Ki = 12900 nM T12808 C5BEZ8 392223 IC50 = 59000 nM T12808 CB9F1O 447961 Ki > 1000 nM T12808 C0G6JH 455733 Ki = 334 nM T12808 C6OAJ7 465908 IC50 > 100000 nM T12808 CK67IQ 465909 IC50 = 68000 nM T12808 CC6Y2M 465910 IC50 > 100000 nM T12808 C9SC7U 465913 IC50 = 40000 nM T12808 CV96KW 465921 IC50 = 22100 nM T12808 CA7J6U 465955 IC50 > 100000 nM T12808 CCG2Y4 465956 IC50 > 100000 nM T12808 CSE5F1 465957 IC50 = 28800 nM T12808 C21DNR 465958 IC50 = 3700 nM T12808 C7GX3E 465959 IC50 > 100000 nM T12808 CW01PD 465961 IC50 > 100000 nM T12808 C1QV3K 465964 IC50 = 78000 nM T12808 CP4V2N 468757 IC50 = 82000 nM T12808 C5UM8B 513197 IC50 = 45300 nM T12808 C1XB9U 637394 IC50 = 1.4 ug.mL-1 T12808 CQ59SY 639665 IC50 > 100000 nM T12808 C6DLK3 644364 IC50 = 3200 nM T12808 C86LNP 2779952 IC50 > 100000 nM T12808 CMKE97 3071991 IC50 > 50000 nM T12808 CTID76 5282335 IC50 > 45000 nM T12808 CY6QK7 5327668 IC50 = 8900 nM T12808 C0J4HV 5327709 IC50 = 6000 nM T12808 C2E5SL 5327711 IC50 = 1900 nM T12808 CSW8K7 5327715 IC50 = 760 nM T12808 C4VTS3 5327723 IC50 = 44700 nM T12808 CNT82G 5327726 IC50 = 20 nM T12808 C6UL3A 5327821 IC50 = 24000 nM T12808 CR3OF4 5327822 IC50 = 24000 nM T12808 C9QMX2 5327823 IC50 = 6900 nM T12808 CA4G1B 5327824 IC50 = 7800 nM T12808 CY2NC3 5327825 IC50 = 5900 nM T12808 CDT07K 5327826 IC50 = 3800 nM T12808 CG36XB 5327827 IC50 = 4700 nM T12808 CF3Y6G 5327828 IC50 = 19000 nM T12808 CY1Z9E 5327829 IC50 > 1000 nM T12808 CI51CH 5327830 IC50 = 4700 nM T12808 CUAW78 5327831 IC50 = 560 nM T12808 CC9US2 5327832 IC50 > 10000 nM T12808 CVGK98 5327833 IC50 > 1000 nM T12808 CGWP86 5327834 IC50 = 2900 nM T12808 C10RVD 5327835 IC50 = 10000 nM T12808 CD6B2A 5327836 IC50 > 10000 nM T12808 CY1O6K 5327837 IC50 > 100000 nM T12808 C1K8CJ 5327838 IC50 > 100000 nM T12808 CP15JO 5327839 IC50 > 10000 nM T12808 CWT9S8 5327840 IC50 > 10000 nM T12808 C5EWD2 5327841 IC50 > 10000 nM T12808 C67JVQ 5327843 IC50 > 10000 nM T12808 CY23QP 5327844 IC50 = 1500 nM T12808 CN1X4Z 5327845 IC50 > 10000 nM T12808 C6TGI1 5327846 IC50 = 3600 nM T12808 CEMR07 5327847 IC50 > 100000 nM T12808 CB90GI 5327848 IC50 = 4500 nM T12808 CLA43B 5327919 IC50 = 270 nM T12808 CPDC54 5327920 IC50 = 5100 nM T12808 CCB9G3 5327921 IC50 = 22 nM T12808 CRTQ98 5327922 IC50 = 40 nM T12808 CP20NQ 5327923 IC50 = 55 nM T12808 C98CNM 5327943 IC50 = 11000 nM T12808 C61URB 5327944 IC50 = 40 nM T12808 CWUY53 5327945 IC50 = 6100 nM T12808 CQ54BE 5327946 IC50 = 110 nM T12808 CIB3P0 5327947 IC50 = 1900 nM T12808 CVG0A1 5327948 IC50 = 210 nM T12808 C8M3PD 5327949 IC50 = 23000 nM T12808 CA25BM 5327950 IC50 = 45000 nM T12808 COP0Q2 5327951 IC50 = 4000 nM T12808 CB47VN 5327952 IC50 = 1900 nM T12808 CPO51K 5327953 IC50 = 410 nM T12808 CI6AY9 5327954 IC50 = 18000 nM T12808 C1Q0PM 5327955 IC50 > 50000 nM T12808 CXA23M 5327956 IC50 = 18000 nM T12808 CH73DT 5327957 IC50 = 3300 nM T12808 CTI6K8 5327963 IC50 = 7800 nM T12808 CAO1N9 5327979 IC50 = 460 nM T12808 CMP3X8 5327994 IC50 = 100 nM T12808 C4DG8Y 5327995 IC50 = 450 nM T12808 CDL0S2 5327996 IC50 > 50000 nM T12808 CC43JH 5327997 IC50 > 50000 nM T12808 CKS8M6 5327998 IC50 = 340 nM T12808 CQ7OZ6 5327999 IC50 = 3600 nM T12808 CQWO93 5328000 IC50 = 11000 nM T12808 CU73IX 5328002 IC50 = 250 nM T12808 CTVP40 5328003 IC50 = 2200 nM T12808 CBSP34 5328004 IC50 = 3100 nM T12808 CS78OD 5328005 IC50 = 19000 nM T12808 CO9YQ6 5328006 IC50 = 17000 nM T12808 CVX2L3 5328007 IC50 = 160 nM T12808 CPD1U9 5328008 IC50 = 130 nM T12808 C3X6QJ 5328012 IC50 = 920 nM T12808 CZO4E1 5328013 IC50 = 4700 nM T12808 C2RA4O 5352033 Ki = 0.26 nM T12808 C7VZ3B 5470616 Ki = 19 nM T12808 C3FY5I 5470617 Ki = 5.9 nM T12808 CJS98K 5470618 Ki = 11 nM T12808 CU7NG8 5470619 Ki = 2.3 nM T12808 CGQ20N 5470620 Ki = 7.3 nM T12808 C2CDY5 5470621 Ki = 5.5 nM T12808 CWP26L 5470622 Ki = 13 nM T12808 C4C3ZX 5470623 Ki = 2.89 nM T12808 CV1T0J 5470624 Ki = 2.7 nM T12808 CF30KU 5470625 Ki = 9 nM T12808 CAP38U 5470626 Ki = 14 nM T12808 C2AUE1 5470627 Ki = 5 nM T12808 CCZ56L 5470628 Ki = 9 nM T12808 CML46Y 5470629 Ki = 16 nM T12808 C47NCD 5470630 Ki = 28 nM T12808 CW4T1V 5470631 Ki = 8 nM T12808 C6CP0R 5470632 Ki = 10 nM T12808 C3J1UV 5470633 Ki = 8.32 nM T12808 C93LKY 5470634 Ki = 11.25 nM T12808 C30RQF 5470635 Ki = 11 nM T12808 CT86FO 5471817 Ki = 3.5 nM T12808 CF32UV 5471818 Ki = 2.9 nM T12808 CB6DU1 5480815 IC50 = 43500 nM T12808 CR06IF 5480816 IC50 > 100000 nM T12808 C69MOJ 5480817 IC50 > 100000 nM T12808 CTAC84 5480818 IC50 = 79200 nM T12808 C5FYU2 5480819 IC50 > 100000 nM T12808 CMXW04 5480821 IC50 > 100000 nM T12808 C35OHQ 5480822 IC50 > 100000 nM T12808 CDK3J0 5703619 IC50 = 0.98 nM T12808 CYBG06 6382557 Ki = 9.5 nM T12808 C0Q1FV 6505653 Ki = 87.2 nM T12808 CN37ZA 6520132 Ki = 54 nM T12808 CGAE28 6520133 Ki = 6.6 nM T12808 CDEK51 6520575 Ki = 29.5 nM T12808 CW1ZY2 6520576 Ki = 3.25 nM T12808 CW9S3K 6538900 IC50 = 22000 nM T12808 C31HEX 6539139 IC50 = 13800 nM T12808 CY20RA 7458031 IC50 > 100000 nM T12808 CQ57EC 9548013 IC50 > 100000 nM T12808 CU6RO8 9797309 Ki = 190 nM T12808 CBT0X5 9797847 IC50 = 52750 nM T12808 CZR3M4 9799152 IC50 = 300 nM T12808 C4PA5X 9800852 Ki = 580 nM T12808 CGC5T3 9800963 Ki = 5.42 nM T12808 CI3O6X 9814609 IC50 = 2600 nM T12808 CUNV09 9816954 IC50 > 100000 nM T12808 CX9DG5 9822042 IC50 > 100000 nM T12808 C8J1OL 9826373 IC50 = 300 nM T12808 C34MXO 9828481 Ki = 0.54 nM T12808 CSH0A9 9847014 IC50 = 180 nM T12808 CT3NJ7 9853645 IC50 = 2600 nM T12808 C3UQL7 9860872 IC50 = 790 nM T12808 CCJK12 9865633 Ki = 14.7 nM T12808 CY70OD 9882602 IC50 > 100000 nM T12808 CV1A2S 9883384 IC50 > 100000 nM T12808 C20NKA 9889351 IC50 = 400 nM T12808 CT83AS 9893161 Ki = 83.6 nM T12808 CXA5C8 9893493 IC50 > 50000 nM T12808 C2TC1L 9910609 IC50 > 125000 nM T12808 C1MU0H 9928190 IC50 = 4.6 ug.mL-1 T12808 CQD2W7 9935079 IC50 = 86 nM T12808 COWH06 9935767 Ki = 11.9 nM T12808 CUKH27 9943194 IC50 = 210000 nM T12808 CU78NO 9947433 IC50 = 1700 nM T12808 CYI65J 9948215 IC50 > 100000 nM T12808 CJO47T 9948405 IC50 > 10000 nM T12808 C0TJ2V 9949134 Ki = 60 nM T12808 C0U6EJ 9949448 IC50 = 31500 nM T12808 CP5NJ3 9952970 Ki = 46.6 nM T12808 CYT7R9 9953676 IC50 > 100000 nM T12808 CV34AB 9958125 IC50 = 6000 nM T12808 C5B3DJ 9962496 Ki = 1.56 nM T12808 CJ40GO 9965429 IC50 = 240000 nM T12808 CJ84TX 9977154 IC50 = 4400 nM T12808 CKG5P6 9979315 Ki = 38.7 nM T12808 CS6KX8 9980480 Ki = 24 nM T12808 C2W3AV 9995236 IC50 = 1300 nM T12808 CV8I5X 9999342 IC50 > 10000 nM T12808 CR48TO 10000106 Ki = 18400 nM T12808 C5XU8E 10000872 IC50 = 3600 nM T12808 C57DLH 10001523 IC50 = 4000 nM T12808 CV7Z9Y 10002471 IC50 = 1400 nM T12808 CY65CO 10030073 IC50 = 210 nM T12808 C2UGV9 10030483 IC50 = 6700 nM T12808 CSFT25 10032913 IC50 = 5000 nM T12808 C0G5DK 10039959 IC50 = 45000 nM T12808 C7YD1X 10048045 IC50 > 25000 nM T12808 CV8Z0O 10048676 Ki = 12 nM T12808 CHT5B6 10066610 Ki = 13600 nM T12808 C1JUF8 10073832 IC50 > 50000 nM T12808 CF2UG0 10087009 Ki = 39.9 nM T12808 CC0VB9 10088141 IC50 = 1.6 ug.mL-1 T12808 CTFR48 10091138 Ki = 17 nM T12808 C1MX5C 10092243 Ki = 4.81 nM T12808 C2IBQ4 10097263 IC50 = 1.4 ug.mL-1 T12808 CG7JO8 10099482 IC50 = 3300 nM T12808 C93LPQ 10099652 IC50 = 410 nM T12808 CV7M6R 10101785 Ki = 9.2 nM T12808 C63CFD 10111108 IC50 = 350 nM T12808 CEF8U5 10117705 IC50 = 300 nM T12808 CRT67V 10119173 IC50 = 440 nM T12808 CL42XS 10136330 IC50 = 80000 nM T12808 C2O7ZH 10137972 IC50 = 1.4 nM T12808 CZJI60 10141037 IC50 > 10000 nM T12808 C94WRY 10143231 IC50 > 10000 nM T12808 C76TVG 10143584 IC50 = 1200 nM T12808 CLBD08 10144909 IC50 = 260 nM T12808 CUW34X 10157645 IC50 = 320 nM T12808 C7JP1A 10163439 IC50 = 120 nM T12808 COC30E 10181160 IC50 > 100000 nM T12808 C3QZV8 10184859 IC50 = 150 nM T12808 CJN72C 10185160 IC50 = 220 nM T12808 CJ0R2G 10187378 IC50 = 610 nM T12808 C73LXY 10188021 IC50 = 480 nM T12808 CK7UT9 10188786 IC50 = 320 nM T12808 C5P8JC 10206423 IC50 = 673 nM T12808 CGOT91 10207821 IC50 = 110 nM T12808 CUF0W9 10207822 IC50 = 250 nM T12808 C98TUI 10208507 IC50 = 170 nM T12808 C51SKM 10209082 IC50 = 57 nM T12808 CK72XG 10209108 IC50 = 290 nM T12808 C6WJ0T 10221222 EC50 = 2980000 nM T12808 C8W2HS 10224497 Ki = 45.6 nM T12808 C3VK7T 10229967 IC50 = 290 nM T12808 C5TQ7X 10247543 IC50 > 10000 nM T12808 CC7P0T 10272623 IC50 = 1000 nM T12808 C7SFI1 10296883 IC50 = 2.1 nM T12808 CTXN56 10296960 IC50 = 250 nM T12808 C8RD3V 10301884 IC50 > 10000 nM T12808 CAX9W2 10302405 IC50 = 11 nM T12808 CGI86E 10316132 Ki = 15.1 nM T12808 CNE1H0 10318765 IC50 = 4500 nM T12808 CN28JG 10323743 IC50 > 100000 nM T12808 C1FOA5 10326105 IC50 = 1000 nM T12808 C7N4UG 10339156 Ki = 16900 nM T12808 CFU38G 10363814 Ki = 4580 nM T12808 CPT7G4 10373017 IC50 = 24400 nM T12808 CZD47R 10383657 Ki = 96 nM T12808 CO91QP 10384681 Ki = 28.6 nM T12808 C43MEZ 10385357 Ki = 21000 nM T12808 CX18EG 10387733 IC50 = 117000 nM T12808 CEH41V 10392789 IC50 = 20 nM T12808 C3RBY8 10395226 Ki = 125.8 nM T12808 C87NZG 10404829 Ki = 21 nM T12808 C0U6IP 10409451 Ki = 350 nM T12808 CRVE78 10411641 IC50 = 4700 nM T12808 CP4XB5 10413828 Ki = 12.5 nM T12808 CZ29SB 10415905 IC50 > 100000 nM T12808 CQXJ51 10425978 Ki = 261.5 nM T12808 C7HBP6 10429593 IC50 > 10000 nM T12808 CH7KA0 10440317 IC50 = 2800 nM T12808 CT93AX 10440529 IC50 = 460 nM T12808 C4OG3B 10447648 Ki = 17.3 nM T12808 C1NH2F 10451826 Ki = 31.1 nM T12808 CN1DS6 10452500 Ki = 77.9 nM T12808 C36QRS 10453829 Ki = 870 nM T12808 C0BQI9 10455654 Ki = 11 nM T12808 C10PAC 10460251 IC50 = 10 nM T12808 C25LDK 10460643 IC50 > 50000 nM T12808 C2WQ8M 10473563 IC50 > 10000 nM T12808 C1VI3E 10477747 IC50 = 73 nM T12808 C7PLI5 10478569 IC50 > 50000 nM T12808 CMA4J8 10479260 Ki = 674 nM T12808 C93AXD 10481621 IC50 > 100000 nM T12808 CX7S8N 10482293 IC50 = 20 nM T12808 C0EV8B 10494548 IC50 > 100000 nM T12808 C8DH5W 10499619 IC50 > 100000 nM T12808 C78FPR 10501266 IC50 = 290 nM T12808 C76QGP 10506540 IC50 = 50 nM T12808 C2M9KH 10519191 Ki = 359 nM T12808 C47SRT 10522262 Ki = 28000 nM T12808 CKN1C8 10522936 Ki = 12 nM T12808 C50XFM 10522937 Ki = 8.4 nM T12808 CSR8Y5 10527068 IC50 = 1100 nM T12808 CQCM76 10530006 IC50 = 500 nM T12808 CDNP37 10530708 IC50 = 80 nM T12808 C7MLN0 10532807 IC50 = 12000 nM T12808 C6QGD1 10533306 Ki = 188 nM T12808 C5EYJ3 10554684 IC50 = 3000 nM T12808 C71UIS 10555532 IC50 = 9600 nM T12808 CT34EF 10566926 Ki = 409 nM T12808 C8I6DS 10567105 Ki = 138 nM T12808 CW16DN 10568777 IC50 > 100000 nM T12808 CX67AG 10569366 IC50 > 100000 nM T12808 C8EZX2 10572110 Ki = 27300 nM T12808 CNR1V8 10581141 Ki = 118 nM T12808 C8EQK0 10581173 IC50 = 125000 nM T12808 CP8J4O 10590515 IC50 > 100000 nM T12808 CJC31H 10594456 Ki = 1070 nM T12808 CYK54E 10600065 Ki = 19 nM T12808 C50YZW 10604825 IC50 = 52000 nM T12808 CG1A2W 10615027 Ki = 123 nM T12808 C3XS7J 10615186 Ki = 330 nM T12808 C0LHE5 10615400 IC50 > 100000 nM T12808 CX2LV0 10621740 Ki = 10800 nM T12808 C58AYV 10640765 Ki = 51 nM T12808 CD9RS1 10643635 Ki = 35 nM T12808 C54OZL 10645267 Ki = 96 nM T12808 CZ8UA9 10650891 IC50 > 5000 nM T12808 CZ78VR 10660240 IC50 > 100000 nM T12808 C0HU2T 10664884 Ki = 24 nM T12808 CJ1RY9 10667619 Ki = 27200 nM T12808 CJOU71 10671412 IC50 = 240 nM T12808 CM5B6A 10673286 IC50 = 3500 nM T12808 CW2MP1 10676318 IC50 = 630 nM T12808 CAVX96 10686149 IC50 > 500000 nM T12808 CAM6J3 10686569 Ki = 164 nM T12808 C98STY 10691450 Ki = 260 nM T12808 CYK38J 10693142 Ki = 2720 nM T12808 CU6G5Y 10708835 IC50 = 2500 nM T12808 C09KYC 10713291 Ki = 9810 nM T12808 CKU3D8 10714940 Ki = 109 nM T12808 C5QV2E 10718802 Ki = 26 nM T12808 C2L0OS 10719676 Ki = 2380 nM T12808 CZVK65 10729749 IC50 > 100000 nM T12808 CFHO08 10735751 Ki = 68 nM T12808 CFX72K 10738692 Ki = 6510 nM T12808 CROC17 10742646 Ki = 746 nM T12808 CC29OS 10743415 Ki = 1860 nM T12808 CN9I6T 10768377 IC50 = 1800 nM T12808 CL8VH3 10768554 IC50 = 6300 nM T12808 C5YMK8 10769011 IC50 = 20 nM T12808 CL14ZD 10770447 IC50 = 280 nM T12808 C69TBF 10784497 Ki = 138 nM T12808 C1OXH6 10803234 IC50 > 100000 nM T12808 C6I3TE 10810093 Ki = 489 nM T12808 CCPA54 10812851 Ki = 13 nM T12808 C5G2DS 10813848 Ki = 2020 nM T12808 CI4EZ7 10814666 Ki = 580 nM T12808 CH70MQ 10833926 Ki = 10400 nM T12808 C1V5WA 10835508 Ki = 350 nM T12808 C1PRW5 10838593 Ki = 12780 nM T12808 C18MDA 10848423 IC50 > 100000 nM T12808 CBL5R0 10852454 Ki = 390 nM T12808 C27QVU 10854657 Ki = 28 nM T12808 CXHQ70 10860387 Ki = 29.5 nM T12808 C7HPA0 10864309 IC50 = 6000 nM T12808 C1DRE5 10884145 IC50 = 36 ug.mL-1 T12808 C2G5CU 10894726 Ki > 10000 nM T12808 CBU21M 10917131 Ki = 34.2 nM T12808 C1L4ZC 10940039 IC50 = 3800 nM T12808 CMF6Q7 10948218 Ki = 15.1 nM T12808 CQ4WV5 10970282 Ki = 30.1 nM T12808 CSHA14 11014419 Ki = 1260 nM T12808 C57ABS 11025714 Ki = 10430 nM T12808 CR47CD 11025838 Ki = 412 nM T12808 C4QX3R 11026526 Ki = 4.46 nM T12808 C67ICE 11048420 Ki = 6.87 nM T12808 CN5G4X 11068973 Ki = 429.7 nM T12808 CC90KQ 11090231 Ki = 4840 nM T12808 CFU1T0 11131975 Ki = 11 nM T12808 C48HIZ 11155477 IC50 = 250 nM T12808 C67CSJ 11201611 IC50 = 3.7 nM T12808 CUY3X4 11212432 Ki = 1430 nM T12808 CTQW29 11222966 Ki = 44 nM T12808 CH7D3X 11233762 IC50 = 2000 nM T12808 C4ZH3M 11247295 Ki = 55.7 nM T12808 C3ROM0 11247414 IC50 = 0.5 nM T12808 CANY24 11311217 IC50 = 10500 nM T12808 CRZ38O 11315034 IC50 = 136 nM T12808 CF9ZC1 11323800 Ki = 7162 nM T12808 CTLY12 11359830 Ki = 1500 nM T12808 C4ON7Z 11362429 IC50 = 1.8 nM T12808 C3OCV2 11371778 IC50 = 1500 nM T12808 CP7Y2L 11418853 Ki = 62.2 nM T12808 C0APW4 11422034 IC50 > 10000 nM T12808 C7AI2V 11432911 IC50 > 50000 nM T12808 C3EXM4 11440028 IC50 = 1200 nM T12808 C64IGY 11448608 Ki > 5000 nM T12808 C8DNQ2 11453012 IC50 = 300 nM T12808 CJC95A 11454205 IC50 > 10000 nM T12808 C7I6AG 11474111 IC50 = 1300 nM T12808 C6M9NC 11477626 IC50 > 50000 nM T12808 C7RH0J 11487086 Ki = 208 nM T12808 CC70MB 11487087 Ki = 459 nM T12808 CQR05P 11494718 IC50 = 6300 nM T12808 CW26SK 11494919 Ki = 18 nM T12808 CB7Z9N 11495116 Ki = 24 nM T12808 C4KLR9 11502004 Ki = 983 nM T12808 CHT93E 11502159 IC50 = 4800 nM T12808 C7JDK5 11502311 Ki = 36 nM T12808 CZW65P 11502312 Ki = 23 nM T12808 C0GR4C 11502757 Ki = 4.97 nM T12808 CCB7K9 11509646 Ki = 39 nM T12808 CWX5U4 11510117 Ki = 6.04 nM T12808 C4E3XS 11516608 Ki = 14 nM T12808 CA28IK 11516649 Ki = 17 nM T12808 C4YO9P 11516650 Ki = 19 nM T12808 C6TMQ2 11516803 Ki = 6.18 nM T12808 C58EAQ 11523962 Ki = 67 nM T12808 CNQ61U 11524891 IC50 > 10000 nM T12808 CCX3W5 11531194 Ki = 18 nM T12808 CT4XF3 11531366 Ki = 3.78 nM T12808 C3KAC4 11538477 IC50 = 95 nM T12808 C89ILJ 11545267 Ki = 12 nM T12808 C1CD2N 11547825 IC50 = 20 nM T12808 C6FJU5 11560568 IC50 = 400 nM T12808 C9OV5S 11561609 IC50 = 2.7 nM T12808 CUW0C5 11567501 IC50 = 2700 nM T12808 CWRY72 11567821 IC50 = 3200 nM T12808 CZJY10 11574218 Ki = 5874 nM T12808 CD7PF5 11574473 IC50 = 49 nM T12808 C3V1KN 11581499 Ki = 18300 nM T12808 CR8A1Y 11581855 Ki = 14 nM T12808 CYB4V7 11581893 Ki = 22 nM T12808 C1X0QJ 11582185 Ki = 12 nM T12808 CO9KP5 11583459 IC50 > 10000 nM T12808 CPK4S5 11589504 Ki = 73 nM T12808 CTZC27 11589633 Ki = 147 nM T12808 C4WCL9 11603404 IC50 = 2500 nM T12808 CJC95X 11603769 Ki = 9 nM T12808 CA9XJ2 11604381 IC50 = 0.5 nM T12808 C6LDN4 11617898 IC50 = 7200 nM T12808 CI9HQ2 11624816 IC50 = 36 nM T12808 C2LQI8 11624847 Ki = 14290 nM T12808 C1KY0X 11626874 Ki = 6.88 nM T12808 CZE26D 11632515 Ki = 30 nM T12808 C6V4CJ 11632516 Ki = 406 nM T12808 CK34LS 11632737 IC50 > 40000 nM T12808 CZLS19 11632793 Ki = 16 nM T12808 CG60NH 11638724 IC50 = 37500 nM T12808 CQ5S3G 11639520 IC50 = 73 nM T12808 CPM60Q 11639658 Ki = 27 nM T12808 CN9M2I 11646765 Ki = 17 nM T12808 CV2KF5 11646797 Ki = 2400 nM T12808 C7VP5Q 11647098 Ki = 7 nM T12808 C4U3OI 11653515 Ki = 2100 nM T12808 CPZM49 11654084 Ki = 173 nM T12808 C7VLD4 11654176 Ki = 23.7 nM T12808 C8LQP1 11668252 Ki = 670 nM T12808 C6WY5A 11675462 Ki = 43.3 nM T12808 C4XPF2 11676514 Ki = 129 nM T12808 CQ89HM 11682813 Ki = 16.1 nM T12808 C0WHV8 11696960 Ki = 113 nM T12808 C6ERA1 11697079 Ki = 18 nM T12808 CO59MS 11710989 Ki = 28 nM T12808 CGJY80 11710990 Ki = 48 nM T12808 CM2D4Z 11718329 Ki = 6.66 nM T12808 CFJ4I7 11723151 IC50 = 1000 nM T12808 CCX53Q 11729563 IC50 = 200 nM T12808 C7C2FM 11737638 IC50 = 1600 nM T12808 CP7AH3 11755812 IC50 = 50000 nM T12808 C6WX1P 11766978 Ki = 7.8 nM T12808 C91EPU 11797210 Ki = 24 nM T12808 CM10YB 11799388 IC50 = 3500 nM T12808 CP8Y5C 11803489 Ki = 4.82 nM T12808 C0L8QJ 11810893 Ki = 225 nM T12808 CW0YT9 11811028 Ki = 4330 nM T12808 CTN96I 11851810 IC50 = 0.5 nM T12808 CA05OS 11972484 IC50 = 410 nM T12808 CW53JC 11998038 Ki = 110 nM T12808 CK0GN2 12018144 IC50 = 740 nM T12808 C4H7YC 12018155 IC50 = 260 nM T12808 C85RQO 12067104 Ki = 127000 nM T12808 CQ39BY 12115602 IC50 = 2.2 nM T12808 CWUK08 13492269 IC50 = 75000 nM T12808 C2QEX8 13492281 IC50 > 100000 nM T12808 CQ8R2X 14159700 Ki = 3430 nM T12808 C2Z8DQ 14624081 IC50 = 23000 nM T12808 CFI9R3 14707658 IC50 = 8.6 ug.mL-1 T12808 C2SE6X 15119070 Ki = 5300 nM T12808 C9CTD0 15119071 Ki = 31000 nM T12808 C5KD8X 15119072 Ki = 300000 nM T12808 C3YRU7 15295578 IC50 > 50000 nM T12808 C2BX8F 15297223 IC50 = 40 nM T12808 CE04YW 15297224 IC50 = 35000 nM T12808 CZK8V6 16043304 IC50 = 66 nM T12808 C9TU1O 16046126 IC50 > 1000 nM T12808 C7WZY3 16066456 IC50 > 10000 nM T12808 C3UHP1 16110374 Ki = 11.6 nM T12808 CG09SM 16110375 Ki = 15.8 nM T12808 CY61JO 16110376 Ki = 52.7 nM T12808 C9ZG5P 16110377 Ki = 18.3 nM T12808 CE7BI5 16110378 Ki = 15.9 nM T12808 C8UW5J 16110390 Ki = 5.23 nM T12808 C3U9HR 16110391 Ki = 5.88 nM T12808 CJ8G5X 16110392 Ki = 126.9 nM T12808 C10HEA 16110393 Ki = 111.1 nM T12808 C5QVP9 16110394 Ki = 1391 nM T12808 CVZK29 16223008 IC50 > 50000 nM T12808 CC24KI 16667248 IC50 = 490 nM T12808 C0H8UN 16730109 IC50 = 188000 nM T12808 C72THB 16739368 IC50 > 100000 nM T12808 C9BJ7Q 16757577 IC50 = 466000 nM T12808 C8AH1I 17758019 IC50 > 100000 nM T12808 C1GKL6 17758020 IC50 > 40000 nM T12808 CIE58R 17758239 IC50 > 40000 nM T12808 CO6LR5 17758240 IC50 > 40000 nM T12808 CWH37T 17758574 IC50 > 40000 nM T12808 C57NRL 17759787 IC50 > 40000 nM T12808 CFAR38 17814740 IC50 = 662 nM T12808 C3D7WE 17874201 IC50 > 200000 nM T12808 C7CLY0 18780230 IC50 > 30000 nM T12808 C3AZJ2 19037238 IC50 > 200000 nM T12808 C3YER4 19696390 IC50 = 1050 nM T12808 C0WEX3 19966997 IC50 = 850 nM T12808 C25UKC 21081761 IC50 > 30000 nM T12808 CL81VC 21100709 IC50 = 26800 nM T12808 C9AVK0 21113469 IC50 = 98 nM T12808 C3EHM4 21197160 IC50 = 3800 nM T12808 CS15LY 21672114 Ki = 0.4 nM T12808 CJ4G1H 21988178 IC50 = 38500 nM T12808 CH27DF 21988185 IC50 = 78000 nM T12808 COH4Y2 21988214 IC50 = 50000 nM T12808 CZ0X8J 22592015 IC50 > 315 nM T12808 CVR9K4 22907281 IC50 = 340 nM T12808 C0HRM6 22911602 IC50 = 400 nM T12808 CUN67H 23366085 IC50 = 12000 nM T12808 CLG9Z8 23366090 IC50 = 34000 nM T12808 CKYB29 23644745 IC50 = 100 nM T12808 CG6D4M 23647319 IC50 > 10000 nM T12808 CY8Z7X 23647330 IC50 > 10000 nM T12808 C4XD8H 23647348 IC50 > 10000 nM T12808 CFMQ08 24370907 IC50 > 100000 nM T12808 CK73JS 24742033 Ki = 6700 nM T12808 C2UOE0 24766030 IC50 > 50000 nM T12808 CCP2M3 24822704 IC50 > 50000 nM T12808 C43HWQ 24883287 IC50 > 10000 nM T12808 C8DA5Q 24883334 IC50 > 10000 nM T12808 C13QYB 24884503 IC50 > 2000 nM T12808 CY8L7E 24896769 IC50 > 10000 nM T12808 CLZ23U 24951610 IC50 > 30000 nM T12808 C36PKE 24992835 Ki = 428 nM T12808 CMP8Z9 24993483 Ki = 54 nM T12808 CH4RO0 24994728 Ki > 1250 nM T12808 C6E9WR 24995040 Ki = 2650 nM T12808 CS3Q8B 24995659 Ki = 76 nM T12808 C2WXE1 24995663 Ki = 49 nM T12808 C1ONA4 24996161 IC50 = 967 nM T12808 CW38QS 25020248 IC50 = 1000 nM T12808 CY6I9E 25020250 IC50 = 1000 nM T12808 CXJ2H9 25052849 Ki = 13.6 nM T12808 CQNK94 25053046 Ki = 128 nM T12808 C0G1KQ 25053118 Ki = 82.2 nM T12808 C8P3XI 25053263 Ki = 136 nM T12808 C0OI9H 25053465 Ki = 252 nM T12808 C0W2LR 25053469 Ki = 84.7 nM T12808 C6AQE3 25053483 Ki = 212 nM T12808 C4S8GL 25053484 Ki = 86.3 nM T12808 CK5QJ0 25053542 Ki = 1370 nM T12808 C8E5GP 25053543 Ki = 76 nM T12808 CG1QE9 25053544 Ki = 3270 nM T12808 C1NB3R 25053545 Ki = 627 nM T12808 CUEF67 25053546 Ki = 51.9 nM T12808 C0A6HF 25053547 Ki = 78.8 nM T12808 CB6K2Q 25053548 Ki = 177 nM T12808 C8YUR7 25053592 Ki = 343 nM T12808 CX7A0N 25053598 Ki = 12.9 nM T12808 CV1BC9 25053600 Ki = 790 nM T12808 C3Q4FG 25053601 Ki = 1110 nM T12808 CGKE80 25053602 Ki = 33200 nM T12808 CYNQ86 25053603 Ki = 15800 nM T12808 CD89IK 25053657 Ki = 755 nM T12808 CSW45A 25053658 Ki = 174 nM T12808 C5LWM2 25053659 Ki = 27100 nM T12808 CY1FP5 25053660 Ki = 810 nM T12808 C0QCH9 25053661 Ki = 21200 nM T12808 CUSD95 25053662 Ki = 1450 nM T12808 C3ARO8 25053721 Ki = 2940 nM T12808 CYN4W3 25053722 Ki = 144 nM T12808 CLSG15 25053723 Ki = 5100 nM T12808 CFCA73 25053724 Ki = 34100 nM T12808 CN9E5K 25053725 Ki = 4880 nM T12808 CAL60N 25053726 Ki = 25400 nM T12808 C53ZIQ 25053780 Ki = 1020 nM T12808 C9IA3M 25053781 Ki = 150 nM T12808 CAED20 25053782 Ki = 1130 nM T12808 C9FBJ3 25053783 Ki = 132 nM T12808 CC30IS 25053784 Ki = 13.8 nM T12808 CD92FQ 25053849 Ki = 870 nM T12808 C2KY1G 25094210 IC50 > 10000 nM T12808 CDO3X2 25113021 IC50 > 1000 nM T12808 CBI73N 25113026 IC50 > 1000 nM T12808 C1R0JL 25113028 IC50 = 676 nM T12808 C4KL8Q 25113038 IC50 > 1000 nM T12808 CV58WZ 25113039 IC50 = 818 nM T12808 C8KI1Z 25113050 IC50 > 1000 nM T12808 C6BWZ8 25145145 IC50 > 100 nM T12808 C78YWA 25145716 IC50 > 500 nM T12808 C0GL7R 25212179 IC50 = 5800 nM T12808 C87NZS 25212180 IC50 = 5300 nM T12808 CC71QJ 27666048 IC50 > 100000 nM T12808 C2U0NP 30291209 IC50 > 100000 nM T12808 C7S6OT 30291292 IC50 > 100000 nM T12808 C92QDU 42611189 Ki = 465 nM T12808 CW24IK 42633780 Ki = 60 nM T12808 C75GFD 42633960 Ki = 468 nM T12808 C6ND4K 43839983 IC50 > 10000 nM T12808 CG4DJ2 43839997 IC50 > 10000 nM T12808 CD5Z8U 44139091 Ki = 20.8 nM T12808 CAI56R 44139212 Ki = 38 nM T12808 CNX5R1 44139336 Ki = 19.5 nM T12808 CRD90G 44139337 Ki = 6 nM T12808 C9GX5D 44157980 Ki > 3000 nM T12808 CJZ39Q 44157981 Ki = 43 nM T12808 C4UMB7 44158300 Ki = 63 nM T12808 C4G5DI 44158301 Ki = 2400 nM T12808 CLJ8U3 44186531 Ki = 205 nM T12808 CP2WI9 44186749 Ki = 3.2 nM T12808 CK73NR 44219749 IC50 > 50000 nM T12808 C5QFX6 44263382 IC50 = 15 nM T12808 C8RQU2 44263383 IC50 = 7.1 nM T12808 CZG81D 44263384 IC50 = 0.9 nM T12808 C6YRP1 44263385 IC50 = 1502 nM T12808 CZ1UQ4 44268211 Ki = 500 nM T12808 CML4T6 44268258 Ki = 1300 nM T12808 CERY73 44268388 Ki = 200 nM T12808 CZ5CQ2 44268452 Ki = 600 nM T12808 CD8MY0 44268453 Ki = 300 nM T12808 C83QHW 44273476 IC50 > 100000 nM T12808 C8PT0I 44273491 IC50 > 200000 nM T12808 CS6NT3 44273526 IC50 = 55000 nM T12808 CG8H3R 44273527 IC50 = 59000 nM T12808 C7I1NX 44273528 IC50 = 6800 nM T12808 C3EFQ0 44273554 IC50 > 100000 nM T12808 CAJ48G 44273555 IC50 > 100000 nM T12808 C6VYU1 44273559 IC50 = 85000 nM T12808 C1WAE7 44273560 IC50 > 200000 nM T12808 CQEW06 44273561 IC50 > 200000 nM T12808 C82YSI 44273595 IC50 = 71000 nM T12808 CUG08T 44273597 IC50 > 200000 nM T12808 CIC13W 44273598 IC50 > 200000 nM T12808 CC8W2J 44273599 IC50 = 13000 nM T12808 CR1M9A 44273600 IC50 = 65000 nM T12808 CE6F2M 44273605 IC50 = 65000 nM T12808 CBV2Y3 44273617 IC50 = 110000 nM T12808 CAK08Y 44273618 IC50 = 23000 nM T12808 C0HG8U 44273619 IC50 > 100000 nM T12808 CMRX16 44273620 IC50 = 500000 nM T12808 CT79EW 44273623 IC50 > 200000 nM T12808 CZ6SM5 44273624 IC50 > 200000 nM T12808 CA8J9D 44273646 IC50 = 36000 nM T12808 C8JWQ2 44273647 IC50 > 200000 nM T12808 CI72SY 44273652 IC50 = 41000 nM T12808 CB0IL4 44273653 IC50 = 35000 nM T12808 CA6LH1 44273654 IC50 = 130000 nM T12808 C35TZW 44273659 IC50 = 10000 nM T12808 C8U2RI 44273699 IC50 = 12000 nM T12808 CY9LQ3 44273700 IC50 > 200000 nM T12808 C2BNC0 44276054 Ki = 20 nM T12808 CFE07H 44276098 Ki = 27800 nM T12808 C1M2GX 44276131 Ki = 7600 nM T12808 CA73KV 44276139 Ki = 22000 nM T12808 CBCD84 44276141 Ki = 2500 nM T12808 C6OC5Q 44276145 Ki = 7700 nM T12808 C1CTG0 44276150 Ki = 75300 nM T12808 CXY02E 44276164 Ki > 1700000 nM T12808 CTHM93 44276185 Ki = 8700 nM T12808 C63IFO 44276186 Ki = 4100 nM T12808 CAZ52I 44276187 Ki = 187000 nM T12808 CQK7M4 44278002 Ki = 880 nM T12808 CQ13XB 44291629 Ki > 500 nM T12808 CERT91 44291669 Ki > 500 nM T12808 C1FZ6B 44294270 IC50 = 1400 nM T12808 C6A9FK 44294365 IC50 = 22 nM T12808 C4HS3C 44294447 IC50 = 30 nM T12808 CFZ31C 44294493 IC50 = 220 nM T12808 C54GFD 44294623 IC50 = 260 nM T12808 CG89DS 44294661 IC50 = 2200 nM T12808 CE6SI2 44294722 Ki = 90.7 nM T12808 C4XA9T 44294738 Ki = 1040 nM T12808 C1D9JN 44294902 Ki = 823 nM T12808 CEA5R7 44294919 Ki = 320 nM T12808 CIO1L5 44295033 Ki > 500 nM T12808 CAE1C7 44295137 Ki > 500 nM T12808 CLV1J6 44295167 Ki > 500 nM T12808 CG93DH 44295225 Ki > 500 nM T12808 CSHC96 44297347 IC50 = 37000 nM T12808 CYF8O6 44297594 IC50 = 14000 nM T12808 CG1Z2B 44303442 IC50 = 220 nM T12808 CNJ63O 44303517 IC50 = 920 nM T12808 C8RJN7 44303745 IC50 = 3200 nM T12808 CTM59P 44308069 IC50 = 20 nM T12808 CJ4WB9 44308383 IC50 = 50 nM T12808 C1N6SL 44308409 IC50 = 6700 nM T12808 CO83HF 44308467 IC50 = 3300 nM T12808 CYTA85 44308468 IC50 = 9600 nM T12808 C3M4UP 44308469 IC50 = 270 nM T12808 CY4K5F 44308490 IC50 = 74 nM T12808 C7AG9Y 44308609 IC50 = 10 nM T12808 CYN34A 44308610 IC50 = 20 nM T12808 C79WUE 44308611 IC50 = 20 nM T12808 CS63CK 44308612 IC50 = 80 nM T12808 C47BNR 44310732 IC50 = 30 nM T12808 C2ACB1 44310758 IC50 = 40 nM T12808 CXVB19 44310795 IC50 = 2700 nM T12808 CD8OF2 44311036 IC50 = 22 nM T12808 C13TNU 44315122 IC50 = 430 nM T12808 C3YN1R 44315123 IC50 = 1200 nM T12808 CPJ57U 44315124 IC50 = 240 nM T12808 C9HA8T 44315171 IC50 = 40 nM T12808 C2T3VN 44315184 IC50 = 410 nM T12808 C3SP0H 44315423 IC50 = 2200 nM T12808 C8OAE9 44315457 IC50 = 910 nM T12808 C3JS6X 44315503 IC50 = 60 nM T12808 CEZ68T 44315545 IC50 = 540 nM T12808 C73MZU 44322457 IC50 = 31000 nM T12808 C2C3MV 44322458 IC50 = 860 nM T12808 CA4R8N 44322474 IC50 = 43000 nM T12808 C2WUL9 44322520 IC50 = 97000 nM T12808 CU10GA 44322569 IC50 = 500 nM T12808 C3DY4L 44322570 IC50 = 100 nM T12808 C3UMR9 44322571 IC50 = 2200 nM T12808 CE0QG3 44322667 IC50 = 11000 nM T12808 C31QSE 44322668 IC50 = 3600 nM T12808 CIB64S 44322669 IC50 = 7800 nM T12808 C42OZF 44322670 IC50 = 18000 nM T12808 CPL9E5 44322671 IC50 > 5000 nM T12808 C17GFI 44322684 IC50 > 150000 nM T12808 CG2SL8 44322685 IC50 = 460 nM T12808 CU8CK7 44322686 IC50 > 150000 nM T12808 COCR18 44322713 IC50 = 10000 nM T12808 C6DHT8 44322714 IC50 > 150000 nM T12808 CK7CJ9 44322718 IC50 = 34000 nM T12808 C3VA0L 44322719 IC50 = 2600 nM T12808 C6Z9XL 44322720 IC50 > 50000 nM T12808 C8NR7B 44322740 IC50 = 37000 nM T12808 C4X3UE 44322741 IC50 > 150000 nM T12808 C1JY5B 44322762 IC50 > 150000 nM T12808 CGK4V2 44322763 IC50 = 67 nM T12808 CP2X6J 44322771 IC50 > 50000 nM T12808 CA27PF 44322772 IC50 = 3700 nM T12808 C4P5HM 44322773 IC50 = 25000 nM T12808 CZ7N8D 44322811 IC50 = 5600 nM T12808 C4J3RI 44322813 IC50 = 340 nM T12808 C7WZ4D 44322814 IC50 > 50000 nM T12808 CYDA76 44322815 IC50 > 50000 nM T12808 CI6R4S 44322889 IC50 > 150000 nM T12808 CP6Q9H 44322954 IC50 > 50000 nM T12808 C48NJC 44322981 IC50 = 430 nM T12808 C6K5TE 44322982 IC50 > 150000 nM T12808 CFMB02 44323003 IC50 > 50000 nM T12808 C8CO0I 44327591 Ki = 28 nM T12808 C7EB6M 44327705 Ki = 6500 nM T12808 CJ0ZP1 44331332 Ki = 122 nM T12808 CT7VE5 44331341 Ki = 540 nM T12808 C7D6BR 44331342 Ki = 540 nM T12808 CZ5PO9 44331350 Ki = 122 nM T12808 CUJ81Y 44331391 Ki = 122 nM T12808 CBT7Q4 44331396 Ki = 122 nM T12808 CEWJ01 44331397 Ki = 540 nM T12808 CVC8G1 44331424 Ki = 540 nM T12808 CLPC42 44334296 IC50 = 770 nM T12808 CF61IT 44334334 IC50 = 570 nM T12808 CH9SF8 44334367 IC50 = 910 nM T12808 C3BFI4 44334443 IC50 = 290 nM T12808 CUI5O8 44338655 Ki = 1.758 nM T12808 C5MQ6U 44338664 Ki = 13 nM T12808 CTQ94X 44338676 Ki = 1000 nM T12808 CYQK34 44338686 Ki = 1.202 nM T12808 COB3Q2 44338687 Ki = 327 nM T12808 C95SHX 44338689 Ki = 1088 nM T12808 CJ2WV9 44338690 Ki = 579 nM T12808 CIX90O 44338696 Ki = 679 nM T12808 CM24FV 44338736 Ki = 499 nM T12808 CM7H4C 44338782 Ki = 96 nM T12808 C06MWN 44338790 Ki = 327 nM T12808 C4HVT5 44338801 Ki = 499 nM T12808 CLBK09 44338802 Ki = 565 nM T12808 C5C7ME 44338836 Ki = 2.9 nM T12808 C3J2WY 44338839 Ki = 24 nM T12808 C21ZWV 44338840 Ki = 2.3 nM T12808 CPG5F1 44338878 Ki = 565 nM T12808 CEP7N6 44339508 Ki = 22.7 nM T12808 COB9I4 44339524 Ki = 43.8 nM T12808 C4VWH5 44339538 Ki = 19.1 nM T12808 C12KEH 44339634 Ki = 48 nM T12808 CU0EO1 44339780 Ki = 25.7 nM T12808 C68EGF 44339785 Ki = 14.1 nM T12808 C71XMP 44339786 Ki = 28 nM T12808 C1KPW4 44342449 Ki = 4979 nM T12808 CO4N1W 44342455 Ki = 7582 nM T12808 C5TI6V 44342456 Ki = 7460 nM T12808 C62YBH 44343595 IC50 > 100000 nM T12808 CGJ18X 44347830 Ki = 15.8 nM T12808 CEW3S1 44347969 Ki = 1970 nM T12808 CEFO49 44347984 Ki = 11.2 nM T12808 CZQD97 44348280 Ki = 5.6 nM T12808 C9X0UI 44350353 Ki = 75.6 nM T12808 COJ73E 44355185 Ki = 0.93 nM T12808 CJDZ92 44359341 Ki = 11 nM T12808 CU4E9A 44359443 Ki = 13 nM T12808 CP4A2Z 44359489 Ki = 12 nM T12808 CRSK10 44359647 Ki = 20 nM T12808 CQC47W 44359729 Ki = 37700 nM T12808 C3YBA9 44364173 IC50 = 170 nM T12808 CIH03D 44366053 IC50 = 18000 nM T12808 C2JA0O 44369473 Ki = 240 nM T12808 C2AGP7 44369474 Ki = 165 nM T12808 C6GZ4J 44372961 Ki = 736 nM T12808 CUY63D 44373050 Ki = 50.4 nM T12808 CO28BT 44376126 Ki = 4.05 nM T12808 CH5E4R 44384352 Ki = 20 nM T12808 C8X0WA 44384580 Ki = 395 nM T12808 CF01AV 44384717 IC50 = 6000 nM T12808 C8YNC3 44385264 IC50 = 38500 nM T12808 CC95JU 44385548 IC50 = 3000 nM T12808 CGQ57L 44386180 IC50 = 70 nM T12808 CI0Y5L 44386181 IC50 = 40 nM T12808 C1W6NC 44386587 IC50 = 22 nM T12808 C0PU3I 44386588 IC50 = 160 nM T12808 C3J6ZO 44386589 IC50 = 290 nM T12808 C4MZI9 44386931 IC50 > 50000 nM T12808 C8B1LV 44394308 IC50 = 726 nM T12808 C4UR6L 44394355 IC50 = 27 nM T12808 C9CX5A 44394369 IC50 = 968 nM T12808 CKCW90 44394463 IC50 = 2157 nM T12808 CA7ZI5 44394482 IC50 = 727 nM T12808 CP9CT3 44394511 IC50 = 2232 nM T12808 CFX48I 44394512 IC50 = 1620 nM T12808 CS83VP 44394536 IC50 = 460 nM T12808 CIY32A 44394554 IC50 = 730 nM T12808 C6EZ8Y 44394557 IC50 = 558 nM T12808 C6VJF9 44403780 Ki = 622 nM T12808 CH0A8W 44408572 Ki = 1.45 nM T12808 CZO78X 44408602 Ki = 21700 nM T12808 CGXQ92 44425746 Ki = 4.74 nM T12808 CUB12D 44449577 IC50 > 50000 nM T12808 C0MXV2 44450803 IC50 = 6100 nM T12808 CY87UN 44456923 Ki = 112 nM T12808 CW0T1S 44456924 Ki = 1090 nM T12808 CS2CV1 44456938 Ki = 85.5 nM T12808 C4WRN5 44541014 IC50 = 50 nM T12808 C3VRO9 44557921 IC50 > 10000 nM T12808 CRBT21 44561669 Ki = 4.6 nM T12808 C0TUS2 44561670 Ki = 14.8 nM T12808 CCL85F 44575073 IC50 > 50000 nM T12808 CJX06P 44575126 IC50 > 50000 nM T12808 CE8FC7 44575127 IC50 > 50000 nM T12808 C9KG2I 44581261 IC50 = 48300 nM T12808 C5TBY3 44581605 IC50 = 38700 nM T12808 CEX34T 44581606 IC50 = 4100 nM T12808 COY57J 44592504 IC50 = 40 nM T12808 C28QLM 44605035 IC50 > 50000 nM T12808 C75XHS 44605037 IC50 > 50000 nM T12808 CI7MN3 44621943 Ki = 1230 nM T12808 C1V6TC 44622679 Ki > 1250 nM T12808 C96BNW 46179972 IC50 = 1300 nM T12808 C5RUB7 46216774 Ki = 4.4 nM T12808 CQ3RM2 46216775 Ki = 5 nM T12808 CPZ67X 46230921 Ki = 7.83 nM T12808 CNXB47 46230922 Ki = 7.15 nM T12808 CIV2Y5 46230923 Ki = 191 nM T12808 CVYA74 46230924 Ki = 8.2 nM T12808 CVB1O0 46230972 Ki = 8.1 nM T12808 CZ12TE 46230973 Ki = 198.4 nM T12808 CN6F8J 46231026 Ki = 323 nM T12808 CT0RU9 46231027 Ki = 7.74 nM T12808 CC63GD 46231028 Ki = 10.2 nM T12808 CZY0H9 46231029 Ki = 7.44 nM T12808 CPU3V1 46231030 Ki = 378 nM T12808 CSQ7H3 46231084 Ki = 14.5 nM T12808 C4IPN2 46231085 Ki = 6.4 nM T12808 CMK2J9 46231086 Ki = 8.24 nM T12808 C2ET9K 46231087 Ki = 118 nM T12808 CHO5A3 46231160 Ki = 39.3 nM T12808 C93JWM 46231161 Ki = 30.3 nM T12808 C8HK6S 46231162 Ki = 6.38 nM T12808 CY04WN 46231163 Ki = 11.4 nM T12808 C2KA8C 46231215 Ki = 29.7 nM T12808 CFCY08 46231216 Ki = 533 nM T12808 CW7MS0 46231217 Ki = 6.83 nM T12808 CT5I1M 46231218 Ki = 8 nM T12808 C2VHF6 46231267 Ki = 9.3 nM T12808 C21XYP 46231268 Ki = 10.5 nM T12808 C0XCU6 46231269 Ki = 15.6 nM T12808 CM7WF0 46231270 Ki = 36.4 nM T12808 CF7K5R 46231309 Ki = 8.25 nM T12808 C0HF7D 46231310 Ki = 2.9 nM T12808 CYT37A 46232443 IC50 > 50000 nM T12808 C48ZVW 46232555 IC50 > 50000 nM T12808 CS9B1U 46232556 IC50 > 50000 nM T12808 CO3P0J 46866604 IC50 < 50000 nM T12808 CJOM49 46880136 IC50 = 2460 nM T12808 C26SBC 46880299 IC50 = 4200 nM T12808 CGUK43 46880300 IC50 = 1400 nM T12808 C19QMX 46880301 IC50 = 2900 nM T12808 CIQW73 46880303 IC50 = 1000 nM T12808 CNF9A5 46880334 IC50 = 1400 nM T12808 CUYQ70 46880335 IC50 = 2200 nM T12808 CZ36UN 46880908 IC50 = 5500 nM T12808 CRW97F 46880909 IC50 = 6600 nM T12808 C92JKU 46880910 IC50 = 380 nM T12808 CVJ4K0 46899547 IC50 = 1000 nM T12808 C2B8IC 46899551 IC50 = 1000 nM T12808 CSV5B9 46901859 IC50 = 900 nM T12808 C7YJ2X 46901862 IC50 = 1000 nM T12808 CHSF07 49806372 IC50 > 1000 nM T12808 C5ME3S 49806721 IC50 > 50000 nM T12808 C9L3XR 49838879 IC50 > 40000 nM T12808 CQE9D1 50925411 IC50 = 13 nM T12808 CM42BY 51000510 Ki > 1000000 nM T12808 CAZQ43 51003133 IC50 > 1000 nM T12808 CGB7S6 52920656 IC50 = 95 nM T12808 CXA03W 52920796 IC50 > 100 nM T12808 CHP06V 52948258 Ki = 120 nM T12808 C6OTY5 53251320 IC50 = 10000 nM T12808 CR93CL 53308750 Ki = 198 nM T12808 CE8OY2 53317913 IC50 > 100 nM T12808 CD4H3S 53354074 Ki = 356 nM T12808 CB32QT 53354075 Ki > 1250 nM T12808 C8AB5U 53354478 Ki = 205 nM T12808 CU5G3I 53355992 IC50 = 40350 nM T12808 CM7P3W 53357328 IC50 > 50000 nM T12808 CYB9W4 53358652 Ki > 20000 nM T12808 CSWZ97 53358773 Ki > 20000 nM T12808 CEX95O 53358774 Ki > 20000 nM T12808 C8NA4L 53384644 IC50 > 30000 nM T12808 C71OXL 53388145 IC50 = 24200000 nM T12808 CDL28G 53388146 IC50 > 100000000 nM T12808 CUY9G2 53473663 IC50 = 3.6 nM T12808 CGQ7F8 53473746 IC50 = 3.6 nM T12808 CI1ZG3 53473747 IC50 = 1 nM T12808 C67JHW 53473748 IC50 = 1.7 nM T12808 C7EW6O 53473749 IC50 = 7.5 nM T12808 CPH34R 53473750 IC50 > 316 nM T12808 CWH1D4 53473825 IC50 > 316 nM T12808 CM8K2V 53473826 IC50 = 4.5 nM T12808 C9A8HG 53473827 IC50 = 280 nM T12808 C3A8OT 53473828 IC50 = 235 nM T12808 CLX31Q 53473829 IC50 = 202 nM T12808 C8Y9RE 53473918 IC50 = 8.3 nM T12808 C1XFN0 53473919 IC50 = 8.5 nM T12808 CN34UO 53473920 IC50 = 9.1 nM T12808 C2RE5M 53473921 IC50 = 0.4 nM T12808 C9ZUL0 53473922 IC50 = 6.4 nM T12808 CG6FD5 53474007 IC50 = 11 nM T12808 C0Q7JS 53474008 IC50 = 63 nM T12808 C31WZB 53474009 IC50 = 1.4 nM T12808 CJF1M2 53630890 Ki = 1 nM T12808 C7I2US 54581523 IC50 = 8070 nM T12808 CT5FS8 54581856 Ki = 600 nM T12808 CO9WX0 54582518 IC50 = 4810 nM T12808 CYAG97 54583794 Ki = 2340 nM T12808 C1LO8H 54586381 IC50 = 2685 nM T12808 C9PQ4H 54587726 Ki > 20000 nM T12808 CCM71K 54669828 Ki = 600 nM T12808 C1XS2J 54760383 IC50 = 6700 nM T12808 CNB76L 56643505 IC50 = 829 nM T12808 CIA23U 56665223 EC50 = 5040000 nM T12808 CIM94L 56668847 IC50 > 100000000 nM T12808 C8PK0W 56675716 IC50 > 100000000 nM T12808 C5USP1 57327769 IC50 = 220 nM T12808 CZYM98 57327842 IC50 = 740 nM T12808 CS49KB 57327913 IC50 = 730 nM T12808 CEW5L7 57522817 IC50 > 100000 nM T12808 C4SEH5 57522818 IC50 > 100000 nM T12808 CF8IP6 57522819 IC50 > 100000 nM T12808 CJ56CE 57522820 IC50 > 100000 nM T12808 C3XI2P 57523093 IC50 > 100000 nM T12808 CUH3B5 57523094 IC50 > 100000 nM T12808 C3QF2X 57523095 IC50 > 100000 nM T12808 CP0L8E 57690510 Ki = 1230 nM T12808 CS9E2N 57690531 Ki = 459 nM T12808 C2J9WL 57690545 Ki = 10 nM T12808 CQ0OR2 57690846 Ki = 418 nM T12808 CSP2I8 57690850 Ki > 1250 nM T12808 CAU57Q 57969602 Ki = 57 nM T12808 C1LZI4 57969746 Ki = 1020 nM T12808 CD6ZP3 58009815 IC50 = 2800 nM T12808 CWU1Y3 58009825 IC50 = 2600 nM T12808 C8S6MY 58010054 IC50 = 1300 nM T12808 CVK0G4 58056356 IC50 > 50000 nM T12808 COH41P 58325285 IC50 = 84 nM T12808 CU38PN 58367655 Ki = 459 nM T12808 CI37CQ 58394927 IC50 = 1300 nM T12808 C6KO0G 58395044 IC50 = 1700 nM T12808 C8X6YE 58557497 IC50 = 1700 nM T12808 C6BPR2 58985201 IC50 > 30000 nM T12808 CT3EW2 59292007 IC50 = 130 nM T12808 CJ6ZT2 59332810 IC50 = 378 nM T12808 C1MR8Q 60097495 IC50 > 10000 nM T12808 CNL04P 60155126 Ki = 15 nM T12808 C56PUM 60155209 Ki = 4.7 nM T12808 CWTG65 60199327 Ki = 7.5 nM T12808 C1HSE0 67035086 IC50 = 53 nM T12808 CWI6K5 67035106 IC50 > 10000 nM T12808 CV63UL 67240318 IC50 > 10000 nM T12808 C8I7GC 68293638 IC50 > 10000 nM T12808 CD56XK 68293660 IC50 > 10000 nM T12808 CF39DV 68596931 IC50 = 771 nM T12808 C9XLB3 68597337 IC50 = 433 nM T12808 CMQ58W 68597501 IC50 > 1000 nM T12808 CEZU83 68611347 IC50 > 1000 nM T12808 CJ8G3H 68682755 IC50 = 4.7 nM T12808 CJGH31 70285522 IC50 > 1000 nM T12808 C2XV4Q 70694953 IC50 > 100000 nM T12808 CL1HY5 71212233 IC50 > 100000 nM T12808 CKX52R 71212291 IC50 > 100000 nM T12808 C0T2VB 71212317 IC50 > 100000 nM T12808 C5B8NS 71212337 IC50 > 100000 nM T12808 CSN04E 71212395 IC50 > 100000 nM T12808 C1OCW0 71212403 IC50 > 100000 nM T12808 CBX2I4 71212419 IC50 > 100000 nM T12808 CLS4R3 71212434 IC50 > 100000 nM T12808 CTF8M7 71212446 IC50 > 100000 nM T12808 C2Z8CX 71212514 IC50 > 100000 nM T12808 CBT7L3 71212517 IC50 > 100000 nM T12808 C91HPI 71300299 IC50 > 5000 nM T12808 C6UKD4 71450929 IC50 = 25000 nM T12808 CPZ4F6 71451107 IC50 > 1000 nM T12808 CE1C6J 71452743 IC50 = 137000 nM T12808 C5RKX0 71452928 IC50 > 1000 nM T12808 C4T3LE 71456167 Ki = 679 nM T12808 CLZ67D 71456431 IC50 > 1000 nM T12808 CS89CL 71456432 IC50 > 1000 nM T12808 CIZ7M8 71457965 Ki = 1088 nM T12808 C0EAG9 71457966 Ki = 579 nM T12808 CPIH21 71460129 IC50 > 1000 nM T12808 C69NCX 71461845 IC50 > 1000 nM T12808 C9QB5V 71461846 IC50 > 1000 nM T12808 C6O8KG 71461847 IC50 > 1000 nM T12808 CHY91V 71578307 IC50 > 100000 nM T12808 C0W2KX 71578373 IC50 > 100000 nM T12808 C6TX9R 71578374 IC50 > 100000 nM T12808 C2D1RN 71578375 IC50 > 100000 nM T12808 C73MEW 71578445 IC50 > 100000 nM T12808 C5NH3V 71578446 IC50 > 100000 nM T12808 CC65WU 71578447 IC50 > 100000 nM T12808 CIP6Q2 71578520 IC50 > 100000 nM T12808 CPJ19D 71578658 IC50 > 100000 nM T12808 C5W0GC 71578744 IC50 > 100000 nM T12808 CLZ59B 71578745 IC50 > 100000 nM T12808 C07RPM 71583135 Ki = 549 nM T12808 CIQK36 71583246 Ki = 1240 nM T12808 C4MOE6 71583247 Ki > 1250 nM T12808 CU60JG 71718528 IC50 > 50000 nM T12808 CV70GZ 71728100 Ki = 1 nM T12808 C4OAP2 76285721 IC50 = 1600 nM T12808 CFRU64 76285722 IC50 = 1700 nM T12808 CU80OY 76286333 IC50 = 6900 nM T12808 C7Q0AD 76286479 IC50 = 1800 nM T12808 CZF0N7 76287389 IC50 = 4600 nM T12808 C28STM 76287526 IC50 = 5100 nM T12808 CQT3H7 76320726 Ki = 5.9 nM T12808 CM1YT3 76324374 Ki = 16100 nM T12808 C5YW6A 76327937 Ki = 3.5 nM T12808 CK61HY 85469442 IC50 > 10000 nM T12808 C5S7CW 86072887 IC50 > 10000 nM T12808 CTW6L4 86072888 IC50 > 10000 nM T12808 C0OCM7 86072889 IC50 > 10000 nM T12808 CJB2D6 86072906 IC50 > 10000 nM T12808 C5CD0N 86072920 IC50 > 10000 nM T12808 CS4G0K 86291004 Ki = 17.8 nM T12808 CPG3A5 86302574 IC50 > 30000 nM T12808 C1T9SW 86727297 IC50 = 6600 nM T12808 CFB65P 86727308 IC50 = 2900 nM T12808 C2L4TA 86727318 IC50 = 3000 nM T12808 C06XHV 86727577 IC50 = 310 nM T12808 CNK87H 90219670 IC50 = 4100 nM T12808 C2TW8U 90219704 IC50 = 2200 nM T12808 CGM7O0 90220574 IC50 = 2200 nM T12808 CJ84EU 90220857 IC50 = 450 nM T12808 CXPB19 90644017 Ki = 8.25 nM T12808 C6FO1X 90644018 Ki = 12.9 nM T12808 C0Y8ZK 91933875 IC50 > 10 nM T12808 CAU45T 91971978 IC50 > 30000 nM T12808 CTK8O0 118721284 IC50 = 7100 nM T12808 CYK02G 118721560 IC50 = 9400 nM T12808 CDL8V3 118721561 IC50 = 5400 nM T12808 CTS0Y7 118721562 IC50 > 50000 nM T12808 C58EWT 118721563 IC50 > 50000 nM T12808 CV4O8P 118721564 IC50 = 3000 nM T12808 CE23GF 118725578 Ki = 7.05 nM T12808 CGJ59M 118725630 Ki = 4.33 nM T12808 C9CQ6J 118725631 Ki = 15.4 nM T12808 CKV3Z1 118725632 Ki = 10.2 nM T12808 CWV1H6 118725633 Ki = 16.5 nM T12808 CS63AL 118725634 Ki = 13.2 nM T12808 CMY94J 118725635 Ki = 43.9 nM T12808 CYRA47 118725636 Ki = 30.8 nM T12808 CWB3J2 118725637 Ki = 2.78 nM T12808 CZI2W3 118725638 Ki = 12.6 nM T12808 CT6S2F 118725639 Ki = 8.7 nM T12808 C64AMW 118725640 Ki = 9.8 nM T12808 C5W3SJ 118725641 Ki = 8.31 nM T12808 CC3NO0 118725642 Ki = 7.2 nM T12808 CF3CU5 118725643 Ki = 8.26 nM T12808 CDH1U2 118725644 Ki = 33.1 nM T12808 C1G5IE 118725645 Ki = 26.7 nM T12808 C5JX1Z 118725646 Ki = 31.6 nM T12808 CRP91U 118725647 Ki = 24.5 nM T12808 CQCX41 118737057 IC50 > 10000 nM T12808 CR01OY 122178935 Ki = 21.2 nM T12808 CK0VL8 122178936 Ki = 13.8 nM T12808 CG4JB9 122194654 IC50 = 73900 nM T12808 C2VQW1 134817176 Ki = 127 nM T12808 C2KFH7 135398497 Ki > 2000 nM T12808 CS4OW8 135400873 Ki > 2000 nM T12808 CVJK60 135402835 IC50 = 1850 nM T12808 CW0P1Q 135433657 IC50 = 2539 nM T12808 CFAD48 135611170 Ki > 2000 nM T12808 CYDM01 135891431 IC50 > 10000 nM T12808 CJID74 136013449 IC50 = 18000 nM T12808 C39NGD 136026545 IC50 > 50000 nM T12808 CJ7KN6 136250327 Ki = 56 nM T12808 C1TY6N 137631658 IC50 > 10000 nM T12808 C4P5AE 137631716 Ki = 698 nM T12808 C8U1CL 137632318 IC50 = 3600 nM T12808 CSDJ03 137634374 IC50 > 10000 nM T12808 C7F5LK 137634439 IC50 > 10000 nM T12808 CK5LI2 137634643 IC50 > 10000 nM T12808 CP6Q3K 137634870 IC50 > 10000 nM T12808 C49ENV 137635659 IC50 = 8700 nM T12808 CGF95R 137636716 IC50 = 7400 nM T12808 C0WQ4T 137637877 IC50 > 10000 nM T12808 CUIS85 137638312 IC50 = 5700 nM T12808 C94BQA 137638520 IC50 = 7600 nM T12808 C21SUB 137638899 Ki = 257 nM T12808 CXOK62 137639159 IC50 > 10000 nM T12808 CS05VB 137639624 IC50 = 8300 nM T12808 C8S9CP 137639731 IC50 > 10000 nM T12808 C3S2CY 137639895 IC50 > 10000 nM T12808 CHSJ08 137640349 Ki = 83.1 nM T12808 C12UXT 137640959 IC50 = 63 nM T12808 C1SB6C 137642843 IC50 > 10000 nM T12808 C4MQ5Y 137642906 IC50 > 10000 nM T12808 CPJ26N 137642976 IC50 = 2500 nM T12808 CH15QZ 137643717 IC50 = 3.4 nM T12808 CS0YG3 137644558 IC50 = 1200 nM T12808 CTF39Y 137644968 IC50 = 4800 nM T12808 CVK87P 137645302 IC50 > 10000 nM T12808 C3A9TX 137646224 Ki = 504 nM T12808 CV3XS8 137646260 IC50 > 10000 nM T12808 CX5IK9 137647205 IC50 > 10000 nM T12808 CX5BK1 137647477 IC50 = 2900 nM T12808 CI3F0Q 137647696 IC50 = 7100 nM T12808 CJF3E2 137648687 IC50 > 10000 nM T12808 CW1TJ7 137649466 Ki = 73 nM T12808 CK2PS3 137649977 IC50 = 680 nM T12808 C0F3WD 137650435 IC50 > 10000 nM T12808 C5OC2K 137650510 IC50 = 1100 nM T12808 C1K7RF 137651597 IC50 > 10000 nM T12808 CA46UD 137653406 IC50 > 10000 nM T12808 C7CG5F 137654450 IC50 = 1700 nM T12808 C8R0JP 137654554 IC50 > 10000 nM T12808 C7NO2X 137654557 IC50 = 3300 nM T12808 CGV17I 137654863 IC50 > 10000 nM T12808 CSW4Y2 137655245 IC50 > 10000 nM T12808 C24DNY 137655381 IC50 > 10000 nM T12808 C4W0VL 137656116 IC50 > 10000 nM T12808 CR0QK1 137656838 IC50 = 8300 nM T12808 CJ9KZ2 137657230 IC50 > 10000 nM T12808 CH08TM 137658866 IC50 > 10000 nM T12808 C61FIS 137658873 IC50 > 10000 nM T12808 CS61AX 137659496 IC50 > 100000 nM T12808 C5KX6J 137659805 IC50 > 10000 nM T12808 CUG6N7 137660315 IC50 = 2.8 nM T12808 CF42ZX 137660643 IC50 > 10000 nM T12808 CAS65V 137660703 Ki = 106 nM T12808 CAPY58 137661040 IC50 > 10000 nM T12808 C4RTS3 137661076 Ki = 116 nM T12808 C6QA5D 137661222 IC50 = 63 nM T12808 C49QOZ 138393053 IC50 = 71 nM T12808 C2OCB0 139589936 IC50 = 97 nM T12808 C2W4NJ 139589937 IC50 = 980 nM T12808 CK90DE 139589938 IC50 = 1400 nM T12808 C1OXF6 139589939 IC50 = 3200 nM T12808 C0NCJ7 139589940 IC50 = 1400 nM T12808 CNW73T 139589941 IC50 = 460 nM T12808 C1PVA9 139589942 IC50 = 79 nM T12808 CO73YE 139589944 IC50 = 2100 nM T12808 C6VB3O 145925651 IC50 >= 5000 nM T12808 C7ELX9 145949146 Ki = 2308 nM T12808 CZO0S7 145949469 Ki = 25.2 nM T12808 CG1V9D 145949968 Ki = 30.1 nM T12808 CS75PX 145950212 Ki = 28.77 nM T12808 CVY36T 145951556 Ki = 249 nM T12808 CDM0F1 145951838 Ki = 3640 nM T12808 CE1WI4 145951934 Ki = 30.4 nM T12808 CEX16N 145951949 Ki = 37 nM T12808 CHB38K 145953902 Ki = 146 nM T12808 C8MCT0 145954310 Ki = 135 nM T12808 CDQU92 145954325 Ki = 25.4 nM T12808 CY0ID9 145954400 Ki > 30000 nM T12808 CKL8B4 145954900 Ki = 375 nM T12808 C4HP0N 145955235 Ki = 183.8 nM T12808 CK9IQ0 145955940 Ki = 15.6 nM T12808 C0G9KP 145956414 Ki = 25.65 nM T12808 CMRB05 145956847 Ki = 62.5 nM T12808 CYD17P 145957502 Ki = 65.9 nM T12808 CS60UE 145957652 Ki = 42.3 nM T12808 CVK9L5 145958383 Ki = 439 nM T12808 C8UQB9 145958537 Ki = 112 nM T12808 CHFN64 145958744 Ki = 72 nM T12808 CTK58B 145959420 Ki = 79.1 nM T12808 CFWM04 145959424 Ki = 31.3 nM T12808 CQ7S6Z 145959564 Ki > 30000 nM T12808 C0U5CQ 145961000 Ki = 114 nM T12808 C9IY7P 145964008 IC50 = 64 nM T12808 C4ZU2L 145965049 IC50 = 350 nM T12808 CIQ70O 145966247 IC50 = 430 nM T12808 CPH9E3 145967023 IC50 = 280 nM T12808 C2TMZ3 145967445 IC50 = 45 nM T12808 CDNC31 145967951 IC50 > 500 nM T12808 CXS3W4 145971204 Ki = 27.6 nM T12808 C3PO1Q 145971398 IC50 = 110 nM T12808 C94NTF 145971693 Ki = 29 nM T12808 CMXU60 145972550 IC50 = 380 nM T12808 C98QCL 145974536 Ki = 383 nM T12808 C53VBI 145974831 IC50 = 1400 nM T12808 C4FP9E 145975243 IC50 = 250 nM T12808 CMH8Q5 145975400 IC50 = 140 nM T12808 C5V0AH 145977027 IC50 = 2500 nM T12808 C1QY5N 145977386 IC50 = 340 nM T12808 CP97BA 145982455 IC50 = 92 nM T12808 C2MD1Q 155513187 IC50 > 10000 nM T12808 CU34OH 155567589 Ki = 286 nM T12808 D01YWE 25207521 IC50 = 33600 nM T12808 D02KPV 37783 Ki = 0.2 nM T12808 D02XHC 448912 IC50 > 100000 nM T12808 D03MUZ 17759555 IC50 = 23400 nM T12808 D04AXH 11574614 Ki > 10000 nM T12808 D05SLL 44186619 Ki = 319 nM T12808 D06HVH 54613583 IC50 = 2200 nM T12808 D06ZCX 10455969 IC50 = 720 nM T12808 D07ANB 148879 Ki = 33 nM T12808 D07OAT 456214 IC50 > 10000 nM T12808 D07TPU 10394343 IC50 = 19000 nM T12808 D08JPU 3501 IC50 = 2.3 nM T12808 D08LYB 5166 IC50 = 83 nM T12808 D09XIL 11396738 IC50 > 125000 nM T12808 D0C9KC 10850934 IC50 > 100000 nM T12808 D0D2FC 2794188 IC50 = 13500 nM T12808 D0D6MH 11617559 IC50 > 13000 nM T12808 D0F0AX 135413546 IC50 = 700 nM T12808 D0G3BJ 44292399 Ki = 0.14 nM T12808 D0H7DQ 6419755 IC50 = 331 nM T12808 D0IR6U 5494425 IC50 = 1200 nM T12808 D0J4NI 44186618 Ki = 661 nM T12808 D0K5ZY 105000 Ki = 10.96 nM T12808 D0L0UY 9986606 IC50 = 14800 nM T12808 D0L8CK 5273566 IC50 = 600 nM T12808 D0L8HO 2399 IC50 = 1599 nM T12808 D0M5FF 5083 IC50 = 33 nM T12808 D0M9QM 5327820 IC50 > 100000 nM T12808 D0ME9B 46868971 IC50 > 10 nM T12808 D0O9NE 5388063 EC50 = 1560000 nM T12808 D0P4JO 5281773 IC50 = 1900 nM T12808 D0TO6S 2396 IC50 = 10 nM T12808 D0U8UK 11677079 IC50 = 8100 nM T12808 D0W7JA 5273567 IC50 = 4600 nM T12808 D0W7TU 947057 IC50 > 50000 nM T12808 D0X2DH 17814743 IC50 = 7233 nM T12808 D0Z7TM 22273644 IC50 > 50000 nM T12808 D0ZH1U 2051 IC50 > 100000 nM T28713 D0R0MW 5329102 IC50 = 16.84 nM T28713 D08UUL 46700756 IC50 = 32.57 nM T28713 D0A5MC 11712649 IC50 = 28000 nM T28713 D0E3TC 44259 IC50 = 6.7 nM T28713 D0FD6D 11751922 IC50 = 140 nM T28713 D0PM7Q 11152667 IC50 < 10 nM T28713 D03BNU 59604787 IC50 > 10000 nM T28713 D0H4GI 10275001 IC50 > 3000 nM T28713 D0T3ME 156422 IC50 = 19000 nM T28713 CHC5I0 2971839 IC50 > 10000 nM T28713 CPOJ12 3078519 IC50 = 10 nM T28713 C2PGU4 9572071 IC50 = 49320 nM T28713 CA3V0T 9572240 IC50 > 100000 nM T28713 C1DJ6B 9572244 IC50 = 81000 nM T28713 C73SQF 9572245 IC50 = 67500 nM T28713 CJR60A 9572531 IC50 = 78750 nM T28713 C7GBL9 9572533 IC50 = 64800 nM T28713 C8P3DE 9572535 IC50 = 83000 nM T28713 C6MU5H 9572537 IC50 = 84400 nM T28713 CXZK43 9572545 IC50 > 100000 nM T28713 CDF2S5 9572547 IC50 = 48500 nM T28713 CXI68F 9572620 IC50 = 90000 nM T28713 CSG4X7 9572624 IC50 > 100000 nM T28713 CIFU15 9572626 IC50 = 59000 nM T28713 CK2I4R 9572632 IC50 > 100000 nM T28713 C7OZ6U 9572657 IC50 = 90500 nM T28713 CU30ZL 9572659 IC50 > 100000 nM T28713 C6NGW1 9572661 IC50 = 69500 nM T28713 CRA10N 9572663 IC50 > 100000 nM T28713 C7J4HC 9572736 IC50 = 96000 nM T28713 C0PZF7 9902666 IC50 = 24 nM T28713 CDOG52 9923564 IC50 = 640 nM T28713 CH20JO 9924991 IC50 = 23 nM T28713 CA0K9W 9925320 IC50 = 290 nM T28713 CG0EO9 9947651 IC50 = 47 nM T28713 CD6VP2 9966580 IC50 = 100 nM T28713 C0R7VZ 9969614 IC50 = 81 nM T28713 CQYV59 10108984 IC50 = 12 nM T28713 CU16PW 10115542 IC50 = 3.4 nM T28713 CL89TN 10132912 IC50 = 410 nM T28713 C3YIS8 10133199 IC50 = 32.4 nM T28713 CLD4C6 10133911 IC50 = 715 nM T28713 C3GZ0U 10134344 IC50 = 9.8 nM T28713 C6KWR2 10135342 IC50 = 13 nM T28713 C41DBP 10136568 IC50 = 12 nM T28713 CS9P8Y 10155700 IC50 = 133 nM T28713 CG4T7Q 10177646 IC50 = 4.4 nM T28713 CQ35JG 10177780 IC50 = 8.2 nM T28713 CW20UQ 10179864 IC50 = 6.6 nM T28713 CQ7O0X 10180876 IC50 = 14 nM T28713 C2HAL4 10181185 IC50 = 4.5 nM T28713 C0R5AX 10215912 IC50 = 22679 nM T28713 CU84XZ 10222496 IC50 = 5.5 nM T28713 CCMR56 10224042 IC50 = 41 nM T28713 C9ZR6P 10269200 IC50 = 250 nM T28713 CWG83C 10271635 IC50 = 31 nM T28713 C8PTZ5 10274172 IC50 = 820 nM T28713 C98VJP 10292206 IC50 = 17 nM T28713 C4FWX5 10292251 IC50 = 77 nM T28713 CPV49N 10293093 IC50 = 12 nM T28713 CHIZ25 11185301 IC50 = 200 nM T28713 CNA1S5 11186968 IC50 = 1400 nM T28713 CKQ9E3 11209127 IC50 = 1900 nM T28713 CL05RI 11219756 IC50 = 200 nM T28713 CF58HX 11236100 IC50 = 55 nM T28713 C9WN4E 11290847 IC50 = 32 nM T28713 CBOP58 11293798 Ki = 5670 nM T28713 CL1GB0 11314309 IC50 > 10000 nM T28713 C26BZX 11362471 Ki > 10000 nM T28713 C57ZJX 11364253 IC50 = 530 nM T28713 CVAF59 11371378 IC50 = 61 nM T28713 C9M3HQ 11381897 IC50 = 6000 nM T28713 CVBD65 11391078 IC50 = 1100 nM T28713 CWXB93 11397177 Ki > 10000 nM T28713 CWM18I 11406175 IC50 = 7 nM T28713 C1WXC5 11417488 IC50 = 2800 nM T28713 CEW71P 11427396 IC50 = 500 nM T28713 C3TE0F 11441679 IC50 > 10000 nM T28713 C0MP5Z 11443510 IC50 = 680 nM T28713 CEK5L9 11443537 IC50 = 18 nM T28713 C60TPG 11450303 IC50 = 930 nM T28713 CK3YI0 11462262 IC50 = 1200 nM T28713 C75ZGR 11495159 IC50 = 292 nM T28713 CH8V1E 11496192 IC50 = 39 nM T28713 CGS6L5 11501187 IC50 = 231 nM T28713 CK5YT8 11503709 IC50 = 52 nM T28713 C4LK3Y 11508557 IC50 = 158 nM T28713 CT17DP 11511483 IC50 = 82 nM T28713 CRPM34 11518511 IC50 = 60 nM T28713 CTRC13 11524000 IC50 = 78 nM T28713 CQES50 11524997 IC50 = 70 nM T28713 C8A3VZ 11532590 IC50 = 45 nM T28713 CIE5D1 11532902 IC50 = 55 nM T28713 CPF6H7 11538128 IC50 = 110 nM T28713 CTG83F 11539329 Ki > 9500 nM T28713 CW6CI8 11547980 IC50 = 180 nM T28713 COE51W 11559383 IC50 = 80 nM T28713 CACS26 11561968 Ki > 2000 nM T28713 C48JVY 11573587 IC50 = 710 nM T28713 CCU02H 11573615 IC50 = 72 nM T28713 C1CY5E 11575815 IC50 = 37 nM T28713 CBSZ28 11576384 IC50 = 61 nM T28713 CK6TJ2 11576419 IC50 = 67 nM T28713 CZ28UI 11576690 IC50 = 74 nM T28713 CJC4O3 11576691 IC50 = 95 nM T28713 CAJ1F5 11580880 IC50 = 176 nM T28713 CMIL86 11590363 Ki > 9500 nM T28713 C6DVH2 11597675 IC50 = 70 nM T28713 CQZ62P 11601801 IC50 = 52 nM T28713 CEF50Y 11602470 IC50 = 710 nM T28713 CB59EG 11609976 IC50 = 233 nM T28713 C5JRC6 11610261 IC50 = 174 nM T28713 CC7AU2 11624189 IC50 = 180 nM T28713 C1EFJ6 11627602 IC50 = 176 nM T28713 CC7K3I 11630978 IC50 = 73 nM T28713 C9T6SC 11640926 Ki > 9500 nM T28713 C08TIB 11642172 IC50 = 157 nM T28713 CKSL10 11649348 IC50 = 114 nM T28713 C0G9CK 11654372 IC50 = 86 nM T28713 C4SNT1 11676846 IC50 = 57 nM T28713 C5QF3U 11682614 IC50 = 140 nM T28713 CJ9KN7 11683817 IC50 > 10000 nM T28713 CU0E8O 11690457 Ki > 2000 nM T28713 C9UB2E 11691280 IC50 = 23 nM T28713 COK4U9 11691284 IC50 = 90 nM T28713 CXB2S8 11691398 IC50 = 14 nM T28713 CPJO52 11703577 IC50 = 100 nM T28713 C76LAT 11704293 IC50 = 109 nM T28713 CK9XI5 11712859 IC50 = 53 nM T28713 CP5DF9 11719440 IC50 = 90 nM T28713 CFPW41 16007116 Ki > 9500 nM T28713 C9TU1O 16046126 IC50 > 1000 nM T28713 CCQ1W9 16099270 IC50 = 34320 nM T28713 CB04TO 16099272 IC50 = 6580 nM T28713 CHQL75 16099330 IC50 = 59000 nM T28713 C4F8DG 16655048 IC50 = 87 nM T28713 C6QH4P 20299668 IC50 > 20000 nM T28713 C1S9ZB 20299672 IC50 > 100000 nM T28713 C1XLM5 24204009 IC50 > 100000 nM T28713 CMU75L 24204554 IC50 > 100000 nM T28713 CSM03X 24204556 IC50 = 65000 nM T28713 CB4Y6K 24204558 IC50 > 100000 nM T28713 C1TR9Z 24205072 IC50 = 78000 nM T28713 C5GS0O 24205074 IC50 = 79000 nM T28713 C7YG1N 24759534 IC50 = 450 nM T28713 C0MO8J 24800837 IC50 > 100000 nM T28713 CZFK08 24821001 IC50 = 2100 nM T28713 CR27XF 24821002 IC50 = 1800 nM T28713 CZ25YH 24821077 IC50 = 2700 nM T28713 CZQ30O 24822077 IC50 = 3000 nM T28713 CUZP05 24901001 IC50 > 20000 nM T28713 CX1HL8 25032704 Ki > 9520 nM T28713 C05OZY 25068614 IC50 = 3400 nM T28713 C49SOH 25068616 IC50 = 28000 nM T28713 CCGD53 25166905 IC50 = 140 nM T28713 CXOV32 25166906 IC50 = 220 nM T28713 C6NGA0 25166907 IC50 = 300 nM T28713 C7I8JF 25167106 IC50 = 310 nM T28713 CRJ6G0 25167107 IC50 = 470 nM T28713 CLM4X1 25167108 IC50 = 420 nM T28713 CIUJ83 25167109 IC50 = 13 nM T28713 CN6JM1 25167110 IC50 = 1000 nM T28713 CD2FU3 25167111 IC50 = 1800 nM T28713 C7K6TZ 25167112 IC50 = 1200 nM T28713 CU85ZQ 25167308 IC50 = 900 nM T28713 CH7OJ6 25221980 IC50 = 11000 nM T28713 CQKH23 25222088 IC50 = 23000 nM T28713 C6SO9B 25222091 IC50 = 16000 nM T28713 CI9P4F 25222092 IC50 = 12000 nM T28713 C75FIT 25222313 IC50 = 10000 nM T28713 CW58XI 25222318 IC50 = 3500 nM T28713 CB9KL2 25222319 IC50 = 13000 nM T28713 CC71QJ 27666048 IC50 > 100000 nM T28713 COPW43 42610049 IC50 = 41000 nM T28713 CPBZ35 42610232 IC50 = 9600 nM T28713 CTCM25 42610483 IC50 = 8600 nM T28713 C3Q4ZI 42610562 IC50 = 38000 nM T28713 CQ3OK0 44182389 IC50 = 6200 nM T28713 C16LJD 44189155 IC50 = 4600 nM T28713 CN8WB9 44189332 IC50 = 41 nM T28713 COU85V 44203745 IC50 = 17000 nM T28713 C3XP0I 44203747 IC50 = 1800 nM T28713 C7R1QT 44203849 IC50 = 84000 nM T28713 CL3UT1 44203854 IC50 = 12000 nM T28713 CJ7AF4 44203948 IC50 > 100000 nM T28713 CFZT40 44203954 IC50 = 44000 nM T28713 CU7R0F 44205165 IC50 > 100000 nM T28713 CG1VH9 44205166 IC50 = 6600 nM T28713 CHQ7R3 44205167 IC50 > 100000 nM T28713 CW4GS7 44221131 IC50 = 7400 nM T28713 C4B5HM 44221133 IC50 = 5900 nM T28713 CH94TA 44246252 IC50 = 74000 nM T28713 C2RD3Q 44409852 IC50 > 10000 nM T28713 C7D9LM 44409853 IC50 = 1540 nM T28713 CC40LX 44409880 IC50 > 10000 nM T28713 CB5C8Y 44409886 IC50 > 10000 nM T28713 C39FSE 44409887 IC50 = 5800 nM T28713 CPJ85G 44409889 IC50 > 10000 nM T28713 CSX1P8 44409893 IC50 = 2000 nM T28713 C1VT7R 44417767 IC50 = 142 nM T28713 CETQ79 44427518 IC50 = 13450 nM T28713 COPG94 44427519 IC50 > 50000 nM T28713 CUVF14 44444439 IC50 = 35 nM T28713 C2R5WV 44445404 IC50 = 460 nM T28713 CCFQ63 44445405 IC50 = 8000 nM T28713 CSNC31 44445406 IC50 = 11000 nM T28713 C2LZH9 44445408 IC50 = 2300 nM T28713 C3RP1Y 44445409 IC50 > 40000 nM T28713 CM92PX 44445410 IC50 = 37000 nM T28713 CA1X2K 44445411 IC50 = 11000 nM T28713 C3L8SJ 44445412 IC50 = 19000 nM T28713 CA84OX 44445414 IC50 = 5000 nM T28713 CFM15P 44445415 IC50 = 19000 nM T28713 C36WVF 44445416 IC50 = 40000 nM T28713 C2UJP5 44445417 IC50 > 40000 nM T28713 C7GT4U 44445418 IC50 = 17000 nM T28713 C8LJS5 44520782 IC50 = 310 nM T28713 CNI56K 44520783 IC50 = 210 nM T28713 CN4R3E 44520784 EC50 = 5000 nM T28713 CN5V6I 44520785 IC50 = 700 nM T28713 CJ1K0O 44525558 IC50 = 270 nM T28713 C3VN1M 45483148 IC50 = 890 nM T28713 CC6X0H 45483156 IC50 = 960 nM T28713 C2Q0PE 45483158 IC50 = 1120 nM T28713 CRLO64 45483160 IC50 = 580 nM T28713 C8XMC7 45483167 IC50 = 610 nM T28713 CYL4E7 45483171 IC50 = 800 nM T28713 CM15ID 45483173 IC50 = 1130 nM T28713 CY3HW5 46224684 IC50 = 44 nM T28713 CJ9W4F 46229795 IC50 = 610 nM T28713 CT94XF 46229842 IC50 = 2400 nM T28713 C3E0KO 46229843 IC50 = 2300 nM T28713 C5GUX8 46229878 IC50 = 4400 nM T28713 CK6M4T 46229879 IC50 > 100000 nM T28713 CIC92F 46229880 IC50 > 100000 nM T28713 CY1T5F 46229881 IC50 > 100000 nM T28713 CSNY57 46229931 IC50 = 9800 nM T28713 CPHN56 46229932 IC50 = 5200 nM T28713 C62VZF 46229933 IC50 = 6700 nM T28713 C0ZSV9 46229934 IC50 = 6100 nM T28713 CV9QJ4 46229935 IC50 = 85000 nM T28713 CXSZ20 46229984 IC50 = 22000 nM T28713 CHE6Z4 46229985 IC50 = 350 nM T28713 CTPI39 46229986 IC50 = 990 nM T28713 C8OD3M 46229987 IC50 = 1100 nM T28713 C09ANB 46229988 IC50 = 680 nM T28713 CXV25Z 46230035 IC50 = 2200 nM T28713 C2AG0X 46230036 IC50 = 2200 nM T28713 CZ8T7S 46230037 IC50 = 1600 nM T28713 CI3P2X 46230038 IC50 = 600 nM T28713 C1FMB7 46230039 IC50 = 1400 nM T28713 CT82YZ 46230040 IC50 = 420 nM T28713 CA30YZ 46230088 IC50 = 1100 nM T28713 C41RWX 46230089 IC50 = 1350 nM T28713 CGZT61 46230090 IC50 = 830 nM T28713 C8OM5V 46230143 IC50 = 2200 nM T28713 CY97GF 46230144 IC50 > 100000 nM T28713 C45QAU 46230145 IC50 > 10000 nM T28713 CL93DC 46230146 IC50 = 17000 nM T28713 CV5UG7 46230182 IC50 = 410 nM T28713 C52AQD 46230183 IC50 = 3600 nM T28713 C2C0MI 46230184 IC50 = 39 nM T28713 CGNX36 46230185 IC50 = 28 nM T28713 CLS29B 46872626 IC50 > 10000 nM T28713 C2O8RZ 46886323 IC50 > 1000 nM T28713 CRXG74 46911674 IC50 = 120 nM T28713 CNI52G 49797813 IC50 = 1700 nM T28713 C2Z6HW 49797814 IC50 = 2200 nM T28713 CNG4E3 49797838 IC50 = 6000 nM T28713 CBHE98 49797871 IC50 = 6800 nM T28713 CO74EX 49797872 IC50 = 15000 nM T28713 CX5L4V 49797873 IC50 = 480 nM T28713 CNT8C4 49867482 IC50 = 1700 nM T28713 CSF93R 53323279 IC50 = 1050 nM T28713 C0SWH5 53348216 IC50 > 40000 nM T28713 C8NA4L 53384644 IC50 > 30000 nM T28713 CVG90B 53389651 IC50 > 10000 nM T28713 CXV2G6 54770686 IC50 > 100000 nM T28713 C0C7JF 54770689 IC50 > 100000 nM T28713 CES4B3 54770691 IC50 = 90000 nM T28713 C6Z2VS 54770693 IC50 = 41300 nM T28713 C3ZVT2 54770915 IC50 = 93500 nM T28713 CZ3C1P 54770917 IC50 > 20000 nM T28713 C1IX4N 54771375 IC50 > 20000 nM T28713 CME94T 54771590 IC50 > 100000 nM T28713 C5GPT9 54771592 IC50 > 100000 nM T28713 CQY26A 54771820 IC50 > 20000 nM T28713 C1TWQ3 54771822 IC50 > 100000 nM T28713 CBOD63 56835089 IC50 > 30000 nM T28713 CR16SD 56947170 IC50 = 2000 nM T28713 CI82KP 57390271 IC50 > 50000 nM T28713 CHU67R 57390273 IC50 = 18850 nM T28713 C38TVB 57391918 IC50 = 12000 nM T28713 CT1ZU3 57391919 IC50 = 19000 nM T28713 CE8T5V 57393795 IC50 = 88500 nM T28713 CM6F0O 57393798 IC50 > 100000 nM T28713 CGU57X 57394413 IC50 > 100000 nM T28713 CD6Y9Z 57395116 IC50 > 30000 nM T28713 C8W6IG 57395117 IC50 > 30000 nM T28713 CT9L8D 57395512 IC50 > 100000 nM T28713 C2VYZ5 57395514 IC50 > 100000 nM T28713 CGU6C4 57395516 IC50 = 77500 nM T28713 C5KS6T 57395518 IC50 > 100000 nM T28713 C81JSP 57395520 IC50 > 100000 nM T28713 CG7S0D 57396882 IC50 > 30000 nM T28713 CQ6Y4G 57397344 IC50 = 56500 nM T28713 C0HQ1R 57399029 IC50 > 100000 nM T28713 CU82DZ 57400761 IC50 > 20000 nM T28713 CF5LW8 57400763 IC50 > 100000 nM T28713 CE60BZ 57402527 IC50 > 100000 nM T28713 CECL89 57402533 IC50 > 100000 nM T28713 CI50KU 58167984 IC50 = 161 nM T28713 CXJ63M 59603829 IC50 = 420 nM T28713 CQEU96 59603842 IC50 = 24 nM T28713 C1MR8Q 60097495 IC50 > 10000 nM T28713 CK6WO0 66552478 IC50 < 10000 nM T28713 CV63UL 67240318 IC50 > 10000 nM T28713 C32TVX 68230798 IC50 = 410 nM T28713 C5DGR9 69036886 IC50 = 2174 nM T28713 C1IEJ2 70789254 IC50 = 41000 nM T28713 C8T7ZP 70789255 IC50 = 13000 nM T28713 CH0B8N 70789756 IC50 > 30000 nM T28713 CKT60L 71455860 Ki = 88 nM T28713 CG2KF6 71462956 IC50 = 3200 nM T28713 CA3O6K 71552696 IC50 > 30000 nM T28713 C1NPL0 71552941 IC50 > 30000 nM T28713 CA4PS8 71552942 IC50 > 30000 nM T28713 C3UA9C 71553011 IC50 = 30000 nM T28713 CEZ15Y 71553012 IC50 = 30000 nM T28713 CVIA91 71553085 IC50 = 30000 nM T28713 C1TR3O 71553152 IC50 = 30000 nM T28713 CDJY72 71568837 IC50 = 3400 nM T28713 C8CAG7 71578921 IC50 > 10000 nM T28713 C1HW4B 89735655 IC50 = 390 nM T28713 CGB54P 101902999 IC50 = 100 nM T28713 CG62HP 101903000 IC50 = 420 nM T28713 C2Y7MH 118733361 IC50 = 160 nM T28713 C5IBZ8 129851326 IC50 = 1700 nM T28713 C0FM1R 130196825 IC50 = 978 nM T28713 CK8R5Y 134145931 IC50 = 60 nM T28713 C2AN7T 134611886 IC50 > 100000 nM T28713 CLSE63 135398512 IC50 = 24 nM T28713 CW0P1Q 135433657 IC50 = 8 nM T28713 C2LSE6 135566381 IC50 = 160 nM T28713 CXW3V2 135566382 IC50 = 9 nM T28713 CW72QO 135580408 IC50 > 100000 nM T28713 CRJ45X 135589980 IC50 > 50000 nM T28713 C0J3BN 135678111 IC50 = 14649 nM T28713 CDQ19X 135921304 IC50 = 1300 nM T28713 C93PMY 135921306 IC50 = 5100 nM T28713 CT6N5O 135921309 IC50 = 920 nM T28713 CYNJ42 135921333 IC50 = 4600 nM T28713 CZV1F2 135921336 IC50 = 60 nM T28713 CPIU46 135921357 IC50 = 70 nM T28713 CZ3X2M 135921361 IC50 = 92 nM T28713 CT3WF6 135921362 IC50 = 1700 nM T28713 C8GU3S 135921380 IC50 = 181 nM T28713 CN8PE1 135921414 IC50 = 201 nM T28713 C6OD2T 135921415 IC50 = 500 nM T28713 CS75RW 135921431 IC50 = 250 nM T28713 CO4HB9 135921450 IC50 = 600 nM T28713 C35LMX 135921456 IC50 = 78 nM T28713 CCSN86 135921457 IC50 = 510 nM T28713 C1JPV8 135921468 IC50 = 70 nM T28713 C6NPJ1 135921474 IC50 = 28 nM T28713 C5ID4X 135921475 IC50 = 12 nM T28713 CR5P4G 135921484 IC50 = 200 nM T28713 CF96QY 135921485 IC50 = 29 nM T28713 C84AKH 135921502 IC50 = 81 nM T28713 C0V8ZL 135921504 IC50 = 2850 nM T28713 C6GZC8 135921505 IC50 = 154 nM T28713 C8SD7O 135921523 IC50 = 460 nM T28713 CL67HX 135921546 IC50 = 11 nM T28713 C8T5ZB 136016456 IC50 = 1300 nM T28713 CA5IK3 136020049 IC50 = 14 nM T28713 C5XIE8 136026041 IC50 = 34000 nM T28713 CD56MA 136030632 IC50 = 30 nM T28713 C9IYG7 136030656 IC50 = 21 nM T28713 CD5N4W 136030657 IC50 = 280 nM T28713 CSJM98 136030658 IC50 = 11 nM T28713 CSMG59 136030690 IC50 = 180 nM T28713 CZRT29 136030731 IC50 = 37 nM T28713 COC4T2 136042307 IC50 = 20 nM T28713 C0F7XG 136042308 IC50 = 14 nM T28713 CG4S3N 136042309 IC50 = 28 nM T28713 CSV49P 136042310 IC50 = 588 nM T28713 CU4FI9 136042311 IC50 = 1526 nM T28713 CF5S9E 136042312 IC50 = 277 nM T28713 CT4VZ5 136042313 IC50 = 156 nM T28713 CQ69XH 136042314 IC50 = 171 nM T28713 C26ESH 136060555 IC50 = 10300 nM T28713 C7ZIF0 136068426 IC50 = 120 nM T28713 C9S4LY 136068463 IC50 = 14 nM T28713 C8DG4N 136068480 IC50 = 5 nM T28713 CC9U6S 136068516 IC50 = 8 nM T28713 C1M6BD 136068537 IC50 = 65 nM T28713 CAQ7C5 136089402 IC50 = 1500 nM T28713 CXMZ02 136089403 IC50 > 100000 nM T28713 CL0E7M 136089404 IC50 = 1690 nM T28713 COI5K4 136089405 IC50 = 860 nM T28713 C0G7LC 136089406 IC50 = 5400 nM T28713 C0PM7I 137634655 IC50 = 14.9 nM T28713 CTZR97 137635721 IC50 = 33.8 nM T28713 CPX15R 137639924 IC50 = 5.5 nM T28713 C7PCV0 137643275 IC50 = 31 nM T28713 CV5F8A 137645673 IC50 = 17.9 nM T28713 C4PHI6 137647228 IC50 = 48.4 nM T28713 C14DBQ 137650479 IC50 = 52.8 nM T28713 CVI51U 137654925 IC50 = 6.9 nM T28713 CDU90E 137656879 IC50 = 33.4 nM T28713 CZI6C5 137658886 IC50 = 32.5 nM T28713 C4MJ8D 138105941 IC50 = 525 nM T28713 C6VB3O 145925651 IC50 >= 5000 nM T28713 CEN6Y2 145949541 IC50 = 34.57 nM T28713 CPW0I5 145949785 IC50 = 27.88 nM T28713 CD2E5L 145950286 IC50 = 5.55 nM T28713 C8QR2U 145950535 IC50 = 33.8 nM T28713 CM4R3A 145950895 IC50 = 46.2 nM T28713 C3ETR2 145952302 IC50 = 12.9 nM T28713 CWH08J 145953076 IC50 = 9.95 nM T28713 CIY16U 145953158 IC50 = 53.2 nM T28713 CB8W4F 145954303 IC50 = 31.82 nM T28713 C3RG2L 145954676 IC50 = 11.13 nM T28713 CMF35R 145955292 IC50 = 48.72 nM T28713 C2SY6G 145955405 IC50 = 25.84 nM T28713 CD8S3T 145955427 IC50 = 65.07 nM T28713 CVU6J0 145955541 IC50 = 46.29 nM T28713 C45LIN 145955619 IC50 = 11.73 nM T28713 CPJ36L 145956174 IC50 = 15.35 nM T28713 CVN18K 145956210 IC50 = 33.4 nM T28713 CKCE05 145956240 IC50 = 43.82 nM T28713 C17ZKT 145956514 IC50 = 29.2 nM T28713 C0XTC1 145957907 IC50 = 28 nM T28713 CBR8H5 145958058 IC50 = 25.8 nM T28713 CSF5P4 145958152 IC50 = 31.55 nM T28713 CEIK62 145958206 IC50 = 32.4 nM T28713 CY0FH2 145958614 IC50 = 5.56 nM T28713 CL04ZN 145959212 IC50 = 35.91 nM T28713 C9J0XE 145959350 IC50 = 41.64 nM T28713 CX2T6C 145961424 IC50 = 35.9 nM T28713 CWO1M8 145971444 IC50 = 41.64 nM T28713 CWPI41 145971526 IC50 = 11.49 nM T28713 CTU17J 145972015 IC50 = 28.08 nM T28713 C2ZQ8K 145973179 IC50 = 27.91 nM T28713 CEY15H 145974313 IC50 = 40.22 nM T28713 C4UVY7 145976455 IC50 = 31 nM T28713 C2MD1Q 155513187 IC50 > 10000 nM T28713 C86HPW 155518524 IC50 = 79000 nM T28713 CZQM57 155554194 IC50 = 1729 nM T28713 D00ERW 44444843 Ki > 5578 nM T28713 D00HVA 11624601 Ki > 9500 nM T28713 D00MLE 11407345 IC50 = 2400 nM T28713 D01WAI 135451156 IC50 = 183 nM T28713 D03DZO 11715767 IC50 = 1100 nM T28713 D09PTP 57325421 IC50 = 29 nM T28713 D0D3AS 11325003 IC50 = 1500 nM T28713 D0D6DH 10125830 IC50 = 21730 nM T28713 D0DH1H 135564841 IC50 = 3 nM T28713 D0EM1C 9969021 IC50 = 15 nM T28713 D0F0AX 135413546 IC50 = 42 nM T28713 D0O6OH 71553154 IC50 = 7970 nM T28713 D0Q3NG 11715520 Ki > 9500 nM T28713 D0S7IE 11658882 Ki > 9500 nM T28713 D0Z2CN 135418335 IC50 = 3000 nM T28713 D0Z8PT 54758482 IC50 > 10000 nM T82624 CS1QX6 125545 EC50 = 410 nM T82624 C1X6PB 10255407 IC50 = 14 nM T82624 CEG5Y0 44375114 EC50 = 130 nM T82624 CFM3G7 46905360 IC50 = 172 nM T82624 D0A0OJ 125004 IC50 = 20000 nM T82624 D0MR1K 439456 IC50 = 4.43 nM T23499 D00JAU 3749 Ki > 0.0001 nM T23499 D04JEE 4946 EC50 > 5011.87 nM T23499 D09TBD 5344 IC50 = 780 nM T23499 D0S7JH 16004692 IC50 = 0.5 nM T23499 D0U4CE 104865 Ki = 6.5 nM T23499 D0X5ZI 6918493 IC50 = 1 nM T23499 D03LAB 9911482 IC50 = 0.08 nM T23499 D09LQK 443289 IC50 = 0.62 nM T23499 D09XLS 107810 IC50 = 5.3 nM T23499 D0AW8E 151174 IC50 = 18 nM T23499 D0H2RJ 6433095 Ki = 0.13 nM T23499 D0LI1C 44469321 IC50 > 30000 nM T23499 D0QG1B 25099191 IC50 = 3.4 nM T23499 D0R7YY 177236 IC50 = 0.8 nM T23499 D0Y6UU 159594 IC50 = 0.034 nM T23499 D0YS1U 10257882 Ki = 9.3 nM T23499 D05OEO 16212950 IC50 = 0.023 nM T23499 D01EDE 5311192 IC50 = 94 nM T23499 D01VUE 122272 Ki = 48 nM T23499 D02HVW 9910224 IC50 = 21 nM T23499 D07YHT 178103 Ki = 1.1 nM T23499 D0B5PU 9843631 Ki = 1.4 nM T23499 D0H0KK 11742628 IC50 = 7.4 nM T23499 D0J2IH 9912992 IC50 = 1.4 nM T23499 D0J5HU 122044 IC50 = 220 nM T23499 D0L3AR 23670447 Ki = 0.17 nM T23499 D0P0DT 123882 IC50 = 0.24 nM T23499 D0S9JH 122149 IC50 = 3500 nM T23499 D0T1RG 216235 Ki = 0.43 nM T23499 D0W6XL 108002 Ki = 0.2 nM T23499 CK0F2T 5340 IC50 = 69000 nM T23499 CPTS80 123883 IC50 = 0.24 nM T23499 CO51ZQ 129432 IC50 > 50000 nM T23499 CN8XG9 156690 Ki = 10 nM T23499 CG6V4H 157574 IC50 = 0.5 nM T23499 C6MRZ0 182140 IC50 = 40000 nM T23499 CLT7A1 197712 Ki = 1 nM T23499 CN01ID 345351 IC50 = 1300 nM T23499 C6JAK2 2802888 IC50 = 220 nM T23499 COY2S6 2809510 IC50 = 6.2 nM T23499 CAWU68 3370402 IC50 = 500 nM T23499 CUSW87 3765218 IC50 = 10000 nM T23499 CNIO83 3795752 IC50 = 280 nM T23499 CM6FP0 3811690 IC50 = 8900 nM T23499 C32WHK 3847484 IC50 = 7943.28 nM T23499 C25GEL 3921421 Ki = 25 nM T23499 CQ36UV 5017966 IC50 = 1584.89 nM T23499 C7CDI5 5018984 IC50 = 1584.89 nM T23499 CTYX34 5122650 Ki = 19 nM T23499 CP1XZ6 5310990 Ki = 63 nM T23499 CMZ69J 6426756 IC50 = 26000 nM T23499 CP1I9X 6433100 Ki = 3.49 nM T23499 C4UJF5 9797546 Ki = 260 nM T23499 CSDO82 9799352 Ki = 520 nM T23499 CUZ05W 9803428 IC50 = 8.3 nM T23499 C1S4LE 9806559 IC50 = 0.17 nM T23499 CL1Q0S 9807200 Ki = 4.2 nM T23499 C3I8FC 9807456 IC50 = 97 nM T23499 CT3NI6 9807691 IC50 = 4.6 nM T23499 CH5D6W 9808545 IC50 = 488 nM T23499 CA1M0Q 9809270 IC50 = 51 nM T23499 CW7DO3 9809919 IC50 = 0.3 nM T23499 C2OHV0 9810190 IC50 = 2.8 nM T23499 CK5R3H 9810400 IC50 = 86 nM T23499 CN2R6T 9810571 IC50 = 261 nM T23499 CTRI53 9811968 IC50 = 140 nM T23499 C5SPK1 9818889 Ki = 8800 nM T23499 CF04WY 9820754 IC50 = 4300 nM T23499 C74IRJ 9821701 IC50 = 2.4 nM T23499 C4JI2K 9822616 Ki = 0.9 nM T23499 CY6HF0 9825494 IC50 = 0.45 nM T23499 CE6D8F 9826741 IC50 = 8.9 nM T23499 CAG43Q 9827093 IC50 = 1.1 nM T23499 C1T8FJ 9829478 IC50 = 2 nM T23499 C5O9JC 9830098 Ki = 6800 nM T23499 CS93GB 9830495 IC50 = 48 nM T23499 CLO82B 9830773 IC50 = 19 nM T23499 CTL39M 9831249 IC50 = 14 nM T23499 C1VP5Q 9831527 IC50 = 1385 nM T23499 CAE70F 9840391 IC50 = 8.3 nM T23499 C5PW0N 9840650 Ki = 900 nM T23499 C8KIE6 9845562 IC50 = 50 nM T23499 C45MZP 9846065 IC50 = 10000 nM T23499 CD7Z8S 9849547 Ki = 0.43 nM T23499 CXS8Q0 9850566 IC50 = 30 nM T23499 CY4ZL7 9852318 IC50 = 0.4 nM T23499 C72WKR 9852624 IC50 = 1591 nM T23499 CMG10J 9853025 IC50 = 587 nM T23499 CR23PL 9853077 IC50 = 64 nM T23499 C57ROU 9853680 IC50 = 1317 nM T23499 CKN2M5 9864017 Ki = 340 nM T23499 CE3C9Z 9865409 Ki = 0.12 nM T23499 CX4G1B 9865706 IC50 = 1200 nM T23499 C8GX0U 9868379 IC50 = 1 nM T23499 CMU3A0 9868637 IC50 = 0.19 nM T23499 C2A5TY 9868822 IC50 = 28 nM T23499 CR4E6U 9869444 IC50 = 47 nM T23499 CZY6C2 9870830 Ki = 0.17 nM T23499 C04NGY 9870959 IC50 = 0.29 nM T23499 CD8UW0 9871561 IC50 = 26 nM T23499 CG7I2Q 9871837 Ki = 5 nM T23499 CDN81J 9873255 IC50 = 50 nM T23499 C60BJE 9874379 IC50 = 1050 nM T23499 CI6CX4 9874557 IC50 = 77 nM T23499 C05FBL 9885296 IC50 = 1995.26 nM T23499 C41CBX 9888574 IC50 = 2.8 nM T23499 CG57RJ 9890440 IC50 = 2.4 nM T23499 CJ4TB6 9894443 IC50 = 1.8 nM T23499 CR4WY5 9894460 Ki = 0.13 nM T23499 CD04YO 9895957 Ki = 1.9 nM T23499 CB0A3I 9896251 IC50 = 24 nM T23499 CT17KX 9897092 IC50 = 5115 nM T23499 C0UCH8 9897583 IC50 = 130 nM T23499 CJ10PX 9897720 IC50 = 15 nM T23499 C72NYE 9909467 IC50 = 1.1 nM T23499 CZ9P6O 9913198 IC50 = 43 nM T23499 CAL58B 9914310 Ki = 0.069 nM T23499 CU8H1Z 9915028 Ki = 0.46 nM T23499 CE17TJ 9915095 IC50 = 12 nM T23499 CQ1ZN4 9915510 IC50 = 0.55 nM T23499 C2Q9GB 9916121 IC50 = 2.2 nM T23499 C94UCB 9916235 IC50 = 0.08 nM T23499 C5D9ZU 9917072 IC50 = 82 nM T23499 C4Z8KR 9917706 IC50 = 22 nM T23499 C2UWJ3 9927658 Ki = 950 nM T23499 CDE9G5 9932004 IC50 = 13 nM T23499 CXH8R2 9934204 Ki = 17000 nM T23499 C5PLX1 9934302 IC50 = 0.04 nM T23499 CE3GU4 9934580 IC50 = 11 nM T23499 CH34SZ 9936145 Ki = 0.039 nM T23499 CHY6M2 9937336 Ki = 0.11 nM T23499 CI3B9H 9938533 Ki = 1.5 nM T23499 C5E1FA 9938571 Ki = 0.0042 nM T23499 CD6CI8 9939238 IC50 = 0.2 nM T23499 COQ6D7 9939960 IC50 = 10 nM T23499 CU2V9A 9949368 Ki = 820 nM T23499 C5LQV8 9953358 Ki = 6 nM T23499 CYNC62 9953821 IC50 > 1000000 nM T23499 C7TWX3 9955200 IC50 = 1.8 nM T23499 CSXQ79 9956918 IC50 = 3.9 nM T23499 CL81WX 9957225 IC50 = 30 nM T23499 C6HL8T 9957883 IC50 = 100 nM T23499 C5VW8U 9958321 Ki = 0.04 nM T23499 C6HLP5 9959298 IC50 = 4.6 nM T23499 C5P2DZ 9961131 IC50 = 140 nM T23499 CTZ12I 9961347 IC50 = 51703 nM T23499 CD12UT 9979632 Ki = 0.9 nM T23499 CDSG04 9980487 IC50 = 700 nM T23499 CO6B1U 9984193 IC50 = 5.4 nM T23499 CEW8J0 9984393 IC50 = 62 nM T23499 C6BC8U 9985001 Ki = 5 nM T23499 CPS68M 10015852 IC50 = 9200 nM T23499 CI36LH 10021240 IC50 = 9800 nM T23499 C6BLV3 10024044 IC50 = 2000 nM T23499 C9CS4P 10027018 IC50 = 400 nM T23499 CU20QS 10029171 IC50 = 1.8 nM T23499 CF47ZI 10033429 IC50 = 40 nM T23499 CGOR41 10033723 EC50 = 6000 nM T23499 C7KB8D 10038537 IC50 = 2500 nM T23499 C97MQH 10043017 IC50 = 5700 nM T23499 C95BSU 10045790 Ki = 43 nM T23499 C3SX8N 10047521 IC50 = 570 nM T23499 CL2D9Y 10056613 EC50 = 17 nM T23499 C69CLY 10070783 IC50 = 430 nM T23499 C2FQS4 10076527 IC50 = 0.69 nM T23499 CS3E1R 10087191 IC50 = 4000 nM T23499 CU4Y3I 10088869 Ki = 5666 nM T23499 C27QDR 10095637 IC50 = 11000 nM T23499 CCQ9E3 10096179 Ki = 2 nM T23499 CRV84C 10100163 IC50 = 2.5 nM T23499 CER7B9 10102342 IC50 = 430 nM T23499 C8RFO9 10102392 EC50 = 580 nM T23499 CW19OH 10114414 IC50 = 0.08 nM T23499 CKX6Y5 10115469 IC50 = 0.09 nM T23499 CS4BZ7 10119105 IC50 = 9.3 nM T23499 C34YZQ 10119327 IC50 = 0.06 nM T23499 CE7HG5 10119517 Ki = 0.02 nM T23499 C6EA9N 10120430 IC50 = 2.4 nM T23499 C1NCD2 10122033 IC50 = 3.2 nM T23499 CHG8V4 10122442 IC50 = 157 nM T23499 CE73TY 10122495 IC50 = 1280 nM T23499 CQ35RE 10122675 IC50 = 14 nM T23499 CGK62Y 10129267 IC50 = 9.4 nM T23499 C6AYB1 10137382 IC50 = 6.6 nM T23499 CH13YM 10138169 IC50 = 18 nM T23499 C7ED3M 10139080 IC50 = 0.14 nM T23499 CS9T6L 10140418 IC50 = 13 nM T23499 CKT17H 10140871 IC50 = 166 nM T23499 CU1FG6 10140965 IC50 = 5.6 nM T23499 C5G3ZB 10143256 IC50 = 0.05 nM T23499 C9DQ8U 10144334 IC50 = 26 nM T23499 C4ZF9E 10144372 IC50 = 53 nM T23499 CDJ2E1 10145418 IC50 = 8 nM T23499 CV39YI 10146305 IC50 = 1 nM T23499 CIL90P 10146377 IC50 = 2 nM T23499 C0XP7T 10146640 IC50 = 1 nM T23499 C6DV9U 10160887 IC50 = 380 nM T23499 CR2X3P 10163744 IC50 = 0.12 nM T23499 CP6S8W 10163956 IC50 = 6.6 nM T23499 C4R9AN 10165809 IC50 = 18 nM T23499 CZW3K1 10165963 IC50 = 0.1 nM T23499 CRJ6U2 10166104 Ki = 55 nM T23499 CYMP81 10166139 IC50 = 6.7 nM T23499 C2H9PB 10166223 IC50 = 0.68 nM T23499 CLT63F 10166543 IC50 = 2.5 nM T23499 CAJ86X 10166561 Ki = 14 nM T23499 C8S2OA 10166981 IC50 = 17 nM T23499 CHS67I 10168195 IC50 = 27 nM T23499 CF9A4T 10168597 IC50 = 21 nM T23499 CG47TJ 10168939 IC50 = 293 nM T23499 CULK04 10182624 IC50 = 0.43 nM T23499 CF4GW0 10183338 IC50 = 0.05 nM T23499 CRQ3M8 10185233 IC50 = 561 nM T23499 CZ5BC9 10185556 IC50 = 0.03 nM T23499 C15RSN 10187261 IC50 = 5.8 nM T23499 CMN3L6 10187313 IC50 = 6 nM T23499 CA84YS 10187997 IC50 = 0.38 nM T23499 CSI1V8 10188517 IC50 = 155 nM T23499 CE9K4V 10189776 IC50 = 139 nM T23499 CZ3QV1 10190108 IC50 = 7 nM T23499 C3RM1T 10195727 IC50 = 97 nM T23499 CW73GD 10205245 IC50 = 3.4 nM T23499 CG53PL 10205429 IC50 = 452 nM T23499 C6X1YJ 10206155 IC50 = 0.06 nM T23499 C78NXS 10206812 IC50 = 1.27 nM T23499 CNHO17 10206855 IC50 = 0.03 nM T23499 CK9T6Q 10208527 Ki = 40 nM T23499 CO91XK 10208674 IC50 = 0.39 nM T23499 CS7K0L 10209324 Ki = 13 nM T23499 C4V8OE 10209814 IC50 = 6.5 nM T23499 CQ5PU8 10210086 IC50 = 5 nM T23499 CX37UN 10210629 IC50 = 0.14 nM T23499 C3W0LP 10211543 IC50 = 196 nM T23499 C17TGP 10211772 IC50 = 18 nM T23499 C4D2OL 10211781 IC50 = 1 nM T23499 C2XQ5M 10212088 IC50 = 13 nM T23499 C1PA3X 10212163 IC50 = 204 nM T23499 CA9IR4 10218058 IC50 = 25 nM T23499 C05NBT 10224228 IC50 = 7.2 nM T23499 C4JN9U 10224745 IC50 = 12 nM T23499 CEH63U 10226215 IC50 = 3 nM T23499 C9E5VZ 10226239 IC50 = 55.9 nM T23499 CM6R9G 10227760 IC50 = 0.02 nM T23499 C38YUR 10228523 IC50 = 0.03 nM T23499 CJU3O5 10228588 IC50 = 0.07 nM T23499 CM9X1P 10230375 IC50 = 339 nM T23499 C2V3IA 10230546 IC50 = 4.6 nM T23499 CHE0D9 10230703 IC50 = 10.2 nM T23499 C5XB6S 10230737 IC50 = 1.1 nM T23499 CA2M7S 10231591 IC50 = 16 nM T23499 C1AQ8P 10233400 IC50 = 12 nM T23499 CRT27P 10240093 IC50 = 14 nM T23499 CYVT16 10244529 IC50 = 2600 nM T23499 CA31LR 10247887 IC50 = 2800 nM T23499 C0V1MY 10265127 IC50 = 6700 nM T23499 CZXR27 10274552 IC50 = 3.3 nM T23499 CV0W4U 10275056 IC50 = 87.3 nM T23499 C9APT6 10277399 IC50 = 0.14 nM T23499 CFI95E 10278217 IC50 = 0.08 nM T23499 CO18IK 10278777 IC50 = 0.29 nM T23499 CGN2Z4 10279940 IC50 = 4.5 nM T23499 C4JY0V 10280278 IC50 = 1.37 nM T23499 C5LC9E 10280531 Ki = 415 nM T23499 CK4A7M 10280562 Ki = 460 nM T23499 C09UWV 10281192 IC50 = 24 nM T23499 C2MYV8 10281573 IC50 = 125 nM T23499 CQG29F 10281606 IC50 = 51 nM T23499 CS4H7T 10281943 IC50 = 13 nM T23499 CQ2DL1 10282008 IC50 = 2.5 nM T23499 CEH24R 10282163 IC50 = 23 nM T23499 C6TO5E 10298354 IC50 = 6.9 nM T23499 C0JRQ8 10299555 IC50 = 0.21 nM T23499 C64KQN 10302118 IC50 = 22 nM T23499 CE8O1S 10303258 IC50 = 3.5 nM T23499 C5FD9N 10303311 IC50 = 7.4 nM T23499 C56YUP 10304227 IC50 = 12 nM T23499 C57EVT 10305181 IC50 = 753 nM T23499 C3IQ9D 10305334 IC50 = 35 nM T23499 CY1O3L 10321290 IC50 = 0.21 nM T23499 C4HD5U 10321341 Ki = 11.3 nM T23499 C3WX7I 10334781 IC50 = 14000 nM T23499 C40ODB 10336018 IC50 = 7800 nM T23499 CYCK82 10336497 IC50 = 160000 nM T23499 CL8T1D 10337668 IC50 = 13000 nM T23499 CH28KO 10338501 IC50 = 880 nM T23499 CZDC58 10342643 IC50 = 12 nM T23499 CV05AX 10344511 IC50 = 53 nM T23499 CL32JM 10344914 IC50 = 0.062 nM T23499 CVBP57 10347080 IC50 = 1.1 nM T23499 CQVP17 10347783 IC50 = 17.2 nM T23499 CNP9A3 10357554 IC50 = 440 nM T23499 CV9W0K 10366278 IC50 = 0.1 nM T23499 CFQ31T 10366742 IC50 = 42.85 nM T23499 CKB78T 10383884 IC50 = 8.1 nM T23499 CVSG67 10385531 IC50 = 2200 nM T23499 CD36GV 10391968 IC50 = 4.1 nM T23499 C60NHB 10392605 IC50 = 8 nM T23499 C1WZ4L 10395969 EC50 = 2700 nM T23499 CEOA37 10407051 Ki = 422 nM T23499 CRJ63P 10410546 IC50 = 190 nM T23499 C2YZ6V 10412464 IC50 = 310 nM T23499 CB24TQ 10426645 IC50 = 580 nM T23499 CJ2Z1I 10429404 IC50 = 6.2 nM T23499 CG3FC5 10432263 Ki = 0.4 nM T23499 C2T8QW 10433234 IC50 = 110 nM T23499 CP50YC 10440821 IC50 = 1100 nM T23499 CO9N4J 10444974 IC50 = 28000 nM T23499 C6IBW8 10449431 IC50 = 6500 nM T23499 CG59VL 10452089 IC50 = 7300 nM T23499 C2FIW7 10453858 Ki = 15 nM T23499 CNOP08 10463627 IC50 = 4 nM T23499 CIB7Q3 10470588 IC50 = 27000 nM T23499 CI6RA9 10475644 IC50 = 10 nM T23499 C4VE7N 10477792 IC50 = 75000 nM T23499 C4R6AL 10478562 IC50 = 1640 nM T23499 CG4SX2 10479787 IC50 = 46 nM T23499 CFY80N 10496523 IC50 = 6309.57 nM T23499 CQFV65 10501279 IC50 = 90 nM T23499 CJ6N8I 10502226 IC50 = 27 nM T23499 CG3PQ2 10502577 IC50 = 43 nM T23499 CA28OV 10503067 IC50 = 35 nM T23499 CTN0R4 10503334 IC50 = 166 nM T23499 CE6O4M 10503525 IC50 = 6.7 nM T23499 CL15XB 10503921 IC50 = 0.63 nM T23499 CVD26B 10503976 IC50 = 1910 nM T23499 CYSG24 10504542 IC50 = 17 nM T23499 C8N3GD 10504689 IC50 = 8.5 nM T23499 CWI0N5 10504920 IC50 = 3.8 nM T23499 C2DFV1 10505209 IC50 = 14 nM T23499 CB31YK 10505357 Ki = 32 nM T23499 CST2V6 10505434 Ki = 23 nM T23499 CJFM87 10506068 IC50 > 25000 nM T23499 CKE8Q4 10506430 IC50 = 200 nM T23499 CC6GL2 10506505 IC50 = 29 nM T23499 CIW27H 10508342 Ki = 290 nM T23499 C1B6NO 10516176 IC50 = 770 nM T23499 CEG80Q 10525281 IC50 = 2.7 nM T23499 COH58N 10526002 IC50 = 40 nM T23499 C4KPF8 10527706 IC50 = 21.3 nM T23499 CPD1A6 10527774 IC50 = 104 nM T23499 CRYH40 10528383 IC50 = 2000 nM T23499 CGL8S2 10528863 Ki = 3.48 nM T23499 C7H8QX 10529868 IC50 = 15 nM T23499 C9VB4O 10530409 IC50 = 0.5 nM T23499 C6VMG1 10531506 IC50 = 122 nM T23499 CZ5XU3 10540843 IC50 = 3800 nM T23499 CN3K9V 10546830 IC50 = 838 nM T23499 C2L5NQ 10548486 IC50 = 32 nM T23499 CH3TX0 10548722 Ki = 3.7 nM T23499 CGJ98W 10549472 Ki = 70 nM T23499 C5PBZ2 10550033 IC50 = 1290 nM T23499 CE0OB4 10550094 IC50 = 630.96 nM T23499 CV60OA 10552007 IC50 = 1300 nM T23499 CL7X5F 10552051 IC50 = 31 nM T23499 CM30IW 10552548 IC50 = 11 nM T23499 C9SW8J 10552683 Ki = 245 nM T23499 C6RH4Q 10553165 IC50 = 950 nM T23499 CDLU05 10553384 IC50 = 1.06 nM T23499 CMW5I1 10553490 IC50 = 5.1 nM T23499 CIE84N 10553793 Ki = 1.5 nM T23499 CBY05M 10554085 IC50 = 19600 nM T23499 CT5JP4 10554384 IC50 = 220 nM T23499 C4BSH1 10554410 IC50 = 41 nM T23499 CUTR43 10554539 IC50 = 6.1 nM T23499 CID50O 10555112 Ki = 1.92 nM T23499 C2BDQ5 10555191 IC50 = 1 nM T23499 CGF3D2 10555208 IC50 = 63.5 nM T23499 C1RS0J 10555424 IC50 = 0.3 nM T23499 CL20OW 10555806 IC50 = 322 nM T23499 CH4KT2 10568280 IC50 = 1000 nM T23499 C6CZ8U 10569313 IC50 = 1584.89 nM T23499 C8GL9N 10575755 IC50 = 27 nM T23499 C29LIN 10575845 IC50 = 15 nM T23499 C49SNK 10576377 IC50 = 85 nM T23499 C69OHR 10576378 IC50 = 132 nM T23499 C7ES1R 10576379 IC50 = 24 nM T23499 CT75CF 10576427 IC50 = 1.2 nM T23499 CLW2T1 10576863 IC50 = 150 nM T23499 C9NS2G 10576888 IC50 = 214 nM T23499 C4C7XI 10576889 IC50 = 62 nM T23499 C38AFS 10577255 IC50 = 200 nM T23499 C0MC2P 10577388 IC50 = 33 nM T23499 CCNG64 10577879 IC50 = 600 nM T23499 C94LZB 10578300 IC50 = 76 nM T23499 CFJ4B1 10578601 IC50 = 22 nM T23499 C8BK7V 10578853 IC50 = 0.2 nM T23499 C8YF3Z 10579100 IC50 = 3.9 nM T23499 CN20UM 10579885 IC50 = 2 nM T23499 C0O3RE 10593411 IC50 = 1258.93 nM T23499 CI52HE 10595728 IC50 = 5011.87 nM T23499 CEM46W 10597575 IC50 = 10 nM T23499 CW4NU5 10599129 Ki = 200 nM T23499 CV69ID 10599230 IC50 = 45.3 nM T23499 CRM76K 10599879 IC50 = 12 nM T23499 CHD87J 10600668 IC50 = 25 nM T23499 CX25TC 10601668 IC50 = 1.8 nM T23499 CM83DC 10602451 IC50 = 680 nM T23499 CKA92J 10602620 IC50 = 15 nM T23499 CK2F0S 10602743 IC50 = 0.9 nM T23499 CN1KQ0 10603135 Ki = 155 nM T23499 C3C6ZP 10603409 IC50 = 0.07 nM T23499 C9YZD4 10604119 IC50 = 27014 nM T23499 C46ZEW 10604167 IC50 = 432 nM T23499 CPEL02 10604797 IC50 = 2000 nM T23499 C3M5OI 10615322 IC50 = 3470 nM T23499 C7GCV1 10621170 IC50 = 57 nM T23499 CSLD54 10622380 IC50 = 30 nM T23499 CR0A3H 10622616 IC50 = 170 nM T23499 C36CFD 10623465 IC50 = 12.59 nM T23499 CK5U1Q 10623757 IC50 = 0.17 nM T23499 CO80EG 10623877 IC50 = 800 nM T23499 C21NHT 10624511 IC50 = 0.1 nM T23499 CY0K7C 10624645 Ki = 32.5 nM T23499 CKZ31J 10625269 IC50 = 25 nM T23499 C7H1BX 10625270 IC50 = 33 nM T23499 CA0C8T 10625694 IC50 = 1 nM T23499 C9QFT0 10625738 IC50 = 977 nM T23499 C74JIT 10626177 IC50 = 470 nM T23499 C4GPV2 10626245 IC50 = 17 nM T23499 CJW2V0 10626362 IC50 = 8.8 nM T23499 C0CR7L 10626646 IC50 = 12 nM T23499 CNQ73U 10627272 IC50 = 0.09 nM T23499 C5XGP4 10627805 IC50 = 61 nM T23499 C5SK8E 10645066 IC50 = 125.89 nM T23499 CB6O1X 10645550 IC50 = 480 nM T23499 CX4F0E 10645779 IC50 = 316.23 nM T23499 C8E5AX 10646372 IC50 = 8 nM T23499 CE0L9G 10646375 IC50 = 240 nM T23499 CF9SD7 10646522 IC50 = 2511.89 nM T23499 C53ANJ 10646616 IC50 = 63.1 nM T23499 CSQR72 10646831 IC50 = 2.6 nM T23499 C3U5HQ 10647021 IC50 = 11 nM T23499 CKP13Z 10647488 IC50 = 22200 nM T23499 CG0H5R 10647642 IC50 = 50 nM T23499 CGE27V 10647898 IC50 = 18 nM T23499 C1TC3P 10648006 IC50 = 0.76 nM T23499 CKEB21 10648937 IC50 = 0.81 nM T23499 CC1G9O 10648996 Ki = 6.03 nM T23499 C6BNY8 10649086 IC50 = 574 nM T23499 C34PRC 10649119 IC50 = 5.5 nM T23499 C32RCS 10650062 IC50 = 9.3 nM T23499 CU25BJ 10650210 IC50 = 4 nM T23499 C43LKS 10650331 IC50 = 450 nM T23499 C5EG7D 10650477 IC50 = 1500 nM T23499 CVJ6M3 10650546 IC50 = 1228 nM T23499 CWH6N0 10651488 IC50 = 0.055 nM T23499 CQM4X9 10665805 IC50 = 320 nM T23499 CI94FC 10667000 IC50 = 7.943 nM T23499 C17DRT 10669224 Ki = 19 nM T23499 C7RE5Y 10670279 IC50 > 25000 nM T23499 CT50AW 10670372 IC50 = 46 nM T23499 CL4BO7 10670600 IC50 = 2.512 nM T23499 CQ7OS0 10670662 Ki = 24 nM T23499 C0XV5H 10671031 Ki = 33 nM T23499 CRQ74D 10671036 IC50 = 13 nM T23499 C6XL4K 10671298 IC50 = 501.19 nM T23499 CCWP21 10671649 IC50 = 16 nM T23499 CXT81R 10671928 IC50 = 10 nM T23499 C85HCL 10672494 IC50 = 20 nM T23499 C3W9OA 10673091 Ki = 19.8 nM T23499 C24AKS 10673756 IC50 = 10 nM T23499 CU36WQ 10673969 IC50 = 21 nM T23499 CGV4O8 10674095 IC50 = 190 nM T23499 CKR7T8 10674176 IC50 = 0.12 nM T23499 CUOS92 10674642 IC50 = 840 nM T23499 CNQW61 10685758 IC50 = 6060 nM T23499 C8KSE6 10690058 IC50 = 1584.89 nM T23499 CK8O3S 10691437 Ki = 18 nM T23499 CG6M7O 10692125 Ki = 130 nM T23499 CPU9X8 10692351 IC50 = 700 nM T23499 CR9SX2 10692649 IC50 = 3162.28 nM T23499 C0GPT3 10693110 IC50 = 630 nM T23499 C2H8OE 10693607 Ki = 7 nM T23499 C87FYW 10694591 IC50 = 1150 nM T23499 CWS8D4 10695071 IC50 = 20 nM T23499 CS1IH0 10695363 IC50 = 3.9 nM T23499 CCQ08V 10696210 IC50 = 10 nM T23499 CW09TH 10696788 IC50 = 88 nM T23499 CC16FS 10697520 IC50 = 3.7 nM T23499 C28DBF 10697633 IC50 = 11 nM T23499 CW6K1Q 10697883 IC50 = 6.8 nM T23499 C0YI4J 10698065 IC50 = 2.5 nM T23499 CZ2G1F 10711546 IC50 = 620 nM T23499 CN5X6J 10715441 IC50 = 27 nM T23499 C2I8XQ 10717504 IC50 = 300 nM T23499 CV64IK 10717923 IC50 = 0.15 nM T23499 CG4JW8 10718141 IC50 = 400 nM T23499 CAJV40 10718688 IC50 = 146 nM T23499 CZJ4P6 10719007 IC50 = 2100 nM T23499 CHPV34 10719157 Ki = 22 nM T23499 C43LWC 10719367 IC50 = 1.7 nM T23499 CQ6S3P 10719598 IC50 = 0.55 nM T23499 CAG5X7 10720982 IC50 = 0.7 nM T23499 C80JTH 10721484 Ki = 250 nM T23499 CQI32K 10722371 IC50 = 0.2 nM T23499 C0K9DB 10722385 IC50 = 0.05 nM T23499 CCD61P 10722389 IC50 = 749 nM T23499 CZA8Y5 10723203 IC50 = 14270 nM T23499 CUZ05E 10740137 IC50 = 1995.26 nM T23499 CJ97NC 10740138 IC50 = 630.96 nM T23499 CC5HL7 10740139 IC50 = 251.19 nM T23499 C6A5TD 10740258 Ki = 11 nM T23499 CIO0Z4 10740439 IC50 = 13 nM T23499 CT8L7G 10740614 IC50 = 500 nM T23499 C3SPZ2 10740942 IC50 = 5011.87 nM T23499 CFA29W 10740943 IC50 = 15.85 nM T23499 CC3OM9 10740953 Ki = 16 nM T23499 CTC6N1 10741025 IC50 = 45 nM T23499 CLT30A 10742005 Ki = 11 nM T23499 C5J6YZ 10742841 IC50 = 14 nM T23499 CGJ2T7 10742968 IC50 = 21000 nM T23499 C48MQX 10743346 Ki = 340 nM T23499 CCA15K 10744040 IC50 = 16 nM T23499 CB74KC 10744085 IC50 = 27 nM T23499 C1SAE7 10745418 IC50 = 920 nM T23499 CI5K1B 10745668 IC50 = 12 nM T23499 C3EYA5 10746431 IC50 = 0.7 nM T23499 CPW0T6 10763862 Ki = 1 nM T23499 CG7WB3 10765057 IC50 = 19 nM T23499 C9WM1S 10765171 IC50 = 70 nM T23499 CVOU41 10766198 IC50 = 229 nM T23499 CCZA72 10766385 IC50 = 8.2 nM T23499 COUL31 10767505 IC50 = 4 nM T23499 CFZ85A 10767778 IC50 = 160 nM T23499 CPTF13 10768897 Ki = 2.37 nM T23499 CAEC98 10768903 IC50 = 1.6 nM T23499 CKWL78 10768904 IC50 = 13.6 nM T23499 C54XWU 10769177 IC50 = 11000 nM T23499 CF0ZA8 10769526 IC50 = 0.29 nM T23499 CULZ60 10769887 Ki = 39.3 nM T23499 CCN2M7 10786696 Ki = 0.7 nM T23499 C25PFC 10786783 IC50 = 1995.26 nM T23499 C9OKT7 10787482 IC50 = 251.19 nM T23499 CLR0N4 10788494 IC50 = 0.97 nM T23499 CBW04Z 10788853 IC50 = 300 nM T23499 CR93VH 10789524 IC50 = 3 nM T23499 CXDC80 10789830 IC50 = 5011.87 nM T23499 CIVE85 10790686 IC50 = 7.5 nM T23499 C86RWA 10790757 IC50 = 1.4 nM T23499 C8W9ZS 10791694 IC50 = 12 nM T23499 C5Q9DW 10792316 IC50 = 100 nM T23499 C4IN2K 10792636 IC50 = 910 nM T23499 CL51IS 10792711 IC50 = 22 nM T23499 C69NMS 10792783 IC50 = 25 nM T23499 C47DXJ 10792934 IC50 = 10 nM T23499 CBM8Y6 10793053 IC50 = 45.9 nM T23499 COUV95 10793160 Ki = 48 nM T23499 CO0MY7 10793187 Ki = 2400 nM T23499 C8P1RH 10805820 IC50 = 1060 nM T23499 CKIV27 10811477 Ki = 4.7 nM T23499 CD15AQ 10811595 IC50 = 15 nM T23499 CCF2R5 10813228 Ki = 2000 nM T23499 CW4MP1 10814036 IC50 = 1.3 nM T23499 CAN8P9 10814297 Ki = 86 nM T23499 CI9Y0N 10814440 IC50 = 2.1 nM T23499 C3KS2I 10814743 IC50 = 123 nM T23499 CO12UX 10814746 IC50 = 14 nM T23499 CIF9U5 10814776 IC50 = 19 nM T23499 C7AV5W 10815005 IC50 = 200 nM T23499 CT2HR0 10815167 IC50 = 54 nM T23499 C9LQ0A 10815168 IC50 = 47 nM T23499 CT5C4K 10815239 Ki = 0.48 nM T23499 CQC01W 10815726 IC50 = 16 nM T23499 CQS3I2 10815823 IC50 = 0.5 nM T23499 CI98CT 10816152 IC50 = 16 nM T23499 CBG9H3 10816667 IC50 = 131 nM T23499 C7R4WU 10816682 IC50 = 2 nM T23499 C6AKY9 10816963 IC50 = 3700 nM T23499 C5B6SE 10817024 IC50 = 199 nM T23499 CF12ET 10818246 IC50 > 10 nM T23499 CH0AC7 10832243 IC50 = 316.23 nM T23499 C7G3DS 10832511 IC50 = 158.49 nM T23499 C1UD8I 10832763 IC50 = 10210 nM T23499 C1JS7N 10833400 IC50 = 398.11 nM T23499 C2TQO1 10833686 IC50 = 740 nM T23499 C7OQ6G 10835335 Ki = 2 nM T23499 CM40OP 10836754 Ki = 174 nM T23499 COTE52 10837085 Ki = 150 nM T23499 CWB28Y 10839533 IC50 = 887 nM T23499 CB67FN 10839618 IC50 = 28 nM T23499 C80GEX 10839947 IC50 = 89 nM T23499 C1LD6J 10840410 IC50 = 8.5 nM T23499 CO4WH7 10840560 Ki = 1.38 nM T23499 CC0OW9 10841170 IC50 = 161 nM T23499 CC3O7N 10841576 IC50 = 100 nM T23499 C8O0PJ 10854399 IC50 = 1090 nM T23499 CCP93B 10864118 Ki = 0.4 nM T23499 CRFU13 10907333 Ki = 0.6 nM T23499 CZ86ML 10918301 Ki = 0.02 nM T23499 CS08OB 10918368 Ki = 0.045 nM T23499 C3ILH7 10929533 Ki = 0.05 nM T23499 CC3JY9 10941084 Ki = 0.009 nM T23499 CD85OB 10941181 Ki = 0.001 nM T23499 CT1X9E 10972867 Ki = 0.2 nM T23499 CME50A 10973161 Ki = 0.15 nM T23499 C5D3ZQ 10973218 Ki = 0.8 nM T23499 CEM41D 10983585 IC50 = 1500 nM T23499 C3RU0A 10984658 Ki = 0.004 nM T23499 C50GTK 11006149 Ki = 6 nM T23499 C3DJP1 11027595 Ki = 0.04 nM T23499 CY0R2V 11027946 IC50 = 0.87 nM T23499 CA26LW 11049336 Ki = 2.5 nM T23499 C84YPI 11059912 Ki = 0.2 nM T23499 CV1N7F 11071062 Ki = 8.5 nM T23499 CA8C6B 11071765 Ki = 0.01 nM T23499 CFP0E7 11081276 Ki = 0.75 nM T23499 CM51RW 11082049 Ki = 0.39 nM T23499 C4T1IB 11082168 Ki = 0.05 nM T23499 C4Q7VR 11103112 Ki = 1 nM T23499 CT2X7H 11103181 Ki = 0.004 nM T23499 CG8AD9 11103326 Ki = 0.15 nM T23499 C91TLO 11113812 Ki = 1.5 nM T23499 CTC76R 11123603 Ki = 0.3 nM T23499 C3Q0LZ 11124425 Ki = 0.02 nM T23499 CY9TE7 11124545 Ki = 0.6 nM T23499 C0KC4B 11124821 Ki = 0.005 nM T23499 CN6R0S 11145758 Ki = 0.005 nM T23499 C2D5QN 11155687 IC50 = 7.3 nM T23499 C53FCK 11156301 IC50 = 58.8 nM T23499 C80CVQ 11156376 IC50 = 45.9 nM T23499 CTGR39 11156692 IC50 = 30.5 nM T23499 CP57YV 11157599 IC50 > 10000 nM T23499 C1X6ON 11167889 IC50 = 3840 nM T23499 C3ZJ8G 11168401 IC50 = 443 nM T23499 C7VD8I 11168474 IC50 = 3.5 nM T23499 CPS0F6 11169125 IC50 = 20.5 nM T23499 CX9KE7 11191999 IC50 = 6.7 nM T23499 C90ZLV 11192437 IC50 > 10000 nM T23499 CN9VF3 11192438 IC50 > 10000 nM T23499 C36ZYQ 11192508 IC50 > 10000 nM T23499 CL5RD9 11202819 IC50 = 604 nM T23499 CUS0J1 11203972 IC50 = 5920 nM T23499 C07BRG 11204331 IC50 = 7.6 nM T23499 C6X3BJ 11224973 IC50 = 20.5 nM T23499 C3ZPJ8 11226740 IC50 = 18.9 nM T23499 CC23LY 11226767 IC50 = 156 nM T23499 CCV95P 11235126 IC50 = 69.8 nM T23499 CG0W4N 11238500 IC50 = 25 nM T23499 CR9CW2 11238540 IC50 = 129 nM T23499 CH6OD0 11273181 IC50 = 104 nM T23499 CZ3IE2 11283571 IC50 = 6.4 nM T23499 CB64EK 11284285 IC50 = 6.3 nM T23499 CX0IP1 11284400 IC50 > 10000 nM T23499 CS87FB 11307120 IC50 = 355 nM T23499 CLR79C 11307457 IC50 = 9.1 nM T23499 C1YK2H 11307805 IC50 = 6.4 nM T23499 CBEW43 11308052 IC50 = 13.9 nM T23499 CBC26X 11318409 IC50 = 5 nM T23499 C8YK9R 11318559 IC50 = 126 nM T23499 C18DIX 11318978 IC50 = 1.4 nM T23499 CAIG09 11330570 IC50 = 7.3 nM T23499 C2N3DR 11330923 IC50 = 18.3 nM T23499 CC35XI 11330927 IC50 = 46.2 nM T23499 C8SL3P 11331242 IC50 = 16.9 nM T23499 CW1OM0 11342005 IC50 = 11.8 nM T23499 C25GKE 11342089 IC50 = 10.2 nM T23499 CM5YT2 11353580 IC50 = 3.1 nM T23499 CS8H7Z 11362537 IC50 = 384 nM T23499 C1BZ2Y 11364770 IC50 = 6.5 nM T23499 CC7X9Q 11365059 IC50 = 17.1 nM T23499 CA58FY 11375934 IC50 = 6.7 nM T23499 C1CZ8A 11376627 IC50 = 9.1 nM T23499 CC0L7O 11377200 IC50 = 7.9 nM T23499 CAN9R5 11385689 IC50 = 605 nM T23499 CY0XU7 11386977 IC50 = 146 nM T23499 CZ7DR0 11387205 IC50 = 112 nM T23499 C5TES2 11387315 IC50 = 221 nM T23499 CY6IN3 11387934 IC50 = 3 nM T23499 C0K7AH 11397857 IC50 = 262 nM T23499 CA2LW1 11398658 IC50 = 7.9 nM T23499 CH41WM 11398818 IC50 = 30.3 nM T23499 CI27JP 11408654 IC50 = 23.4 nM T23499 CZ50YK 11409462 IC50 = 1.47 nM T23499 C8RPX0 11409474 IC50 = 23.7 nM T23499 CL3ZW6 11410074 IC50 = 17.1 nM T23499 C7H1JE 11410410 IC50 = 29 nM T23499 C3PDH6 11421392 IC50 = 3.7 nM T23499 CV62BJ 11421972 IC50 = 11 nM T23499 C7SJ6E 11432418 IC50 = 8.9 nM T23499 CLAI47 11432855 IC50 = 123 nM T23499 CGY8F0 11441050 IC50 = 91.7 nM T23499 C5HNO9 11444738 IC50 = 7.9 nM T23499 C7AY3C 11452452 IC50 = 1570 nM T23499 CZ47BI 11455999 IC50 = 101 nM T23499 CR6SC4 11456110 IC50 = 98.6 nM T23499 C3RX2S 11465096 IC50 = 6600 nM T23499 CH1R6E 11465535 IC50 = 0.14 nM T23499 CF6W3J 11467573 IC50 = 24.9 nM T23499 C61GUD 11477664 IC50 = 7.5 nM T23499 C0V6KP 11478553 IC50 = 7.2 nM T23499 CXSE25 11478911 IC50 = 6.8 nM T23499 CETK86 11488556 IC50 = 927 nM T23499 C79SJN 11489174 IC50 = 83.4 nM T23499 CQM85J 11489318 IC50 = 3.9 nM T23499 CN4BV0 11489946 IC50 = 278 nM T23499 C2R3GN 11490160 IC50 = 102 nM T23499 CKZ29W 11505449 IC50 = 0.7 nM T23499 CQF3S5 11730445 Ki = 0.3 nM T23499 CK9D4G 11731054 Ki = 0.03 nM T23499 CHU05Q 11733544 Ki = 1 nM T23499 C9EF7M 11734435 Ki = 0.44 nM T23499 C29SQH 11744509 IC50 = 110 nM T23499 CU02WN 11751754 IC50 = 2.62 nM T23499 CPS5K7 11752174 IC50 = 387 nM T23499 C2I0XM 11752337 IC50 = 0.04 nM T23499 CX58WI 11753090 IC50 = 17.3 nM T23499 CLWM92 11753582 IC50 = 25.8 nM T23499 CTB8N9 11754273 Ki = 0.2 nM T23499 C2Y0VP 11754394 IC50 = 0.5012 nM T23499 CK0F7T 11757759 IC50 = 0.2 nM T23499 CIP68E 11762890 Ki = 0.07 nM T23499 C8D6ZR 11785180 IC50 = 3950 nM T23499 CRLP96 11785813 IC50 = 5.9 nM T23499 CQE14M 11786120 IC50 = 211 nM T23499 C9VS1O 11792960 IC50 = 1258.93 nM T23499 C0PQ4T 11793037 IC50 = 199.53 nM T23499 CD90NG 11793650 IC50 = 3981.07 nM T23499 CFE86R 11794992 Ki = 0.5 nM T23499 CQ7TL8 11797288 Ki = 19 nM T23499 CTU41I 11797486 IC50 = 56 nM T23499 CE9UG2 11798109 IC50 = 933 nM T23499 C8FX7Z 11798228 IC50 = 70 nM T23499 CUC28M 11798504 IC50 = 4.88 nM T23499 C07UEA 11799541 IC50 = 6 nM T23499 C0CG3O 11799625 IC50 = 50 nM T23499 C7Y5RM 11799973 Ki = 2 nM T23499 CREG48 11799974 Ki = 1.95 nM T23499 CK4ZF6 11800505 IC50 = 310 nM T23499 CTH08J 11800649 Ki = 3.13 nM T23499 C9BF8Z 11800804 IC50 = 1.8 nM T23499 CN4K1R 11801906 Ki = 230 nM T23499 CY0W8I 11812665 Ki = 0.6 nM T23499 CS0ZT2 11813485 Ki = 39 nM T23499 CQ8H3G 11813553 Ki = 0.04 nM T23499 C3U2GJ 11827489 IC50 = 0.76 nM T23499 CFK56Z 12060119 IC50 = 1000 nM T23499 C78LHI 12146375 IC50 = 2750 nM T23499 CO9N0H 13044638 IC50 = 11000 nM T23499 CS2Y5E 14041110 IC50 = 800 nM T23499 CH95CP 14673588 IC50 = 8800 nM T23499 C97HQO 14973488 IC50 = 84000 nM T23499 C6IAF9 14973489 IC50 > 32000 nM T23499 C7C5MB 15289330 IC50 = 20 nM T23499 CH68UI 15289331 IC50 = 86 nM T23499 CYJ51R 15297023 IC50 = 2800 nM T23499 C7MGH2 15297025 IC50 = 1000 nM T23499 CC3RX8 15297287 Ki = 28000 nM T23499 CTZ1E4 15342056 IC50 = 1910 nM T23499 CORE65 15410997 IC50 = 18 nM T23499 C2QA8Y 15411002 IC50 = 9 nM T23499 CC8BP3 15411003 IC50 = 0.8 nM T23499 CC58ZF 15411005 IC50 = 0.6 nM T23499 C2RNU5 15411009 IC50 = 0.5 nM T23499 CGT4Q2 15453170 IC50 = 9900 nM T23499 C1ROV7 15453172 IC50 = 2900 nM T23499 CD7NK1 15453177 IC50 = 1.4 nM T23499 CW0GJ1 15453178 IC50 = 3.8 nM T23499 CJR1T8 15453179 IC50 = 120 nM T23499 C58JIU 15453180 IC50 = 160 nM T23499 CI63TE 15453209 IC50 = 5900 nM T23499 CGHV58 15453210 IC50 = 490 nM T23499 CKM63F 17979733 Ki = 17 nM T23499 C26WMV 17979744 Ki = 1 nM T23499 CM0A3C 17979745 Ki = 55 nM T23499 CHO47W 17979749 Ki = 20 nM T23499 C8NGJ0 18004820 Ki = 40 nM T23499 C52HXB 18184179 IC50 = 2838 nM T23499 C8BGV5 18184194 IC50 = 116 nM T23499 CDU0W6 18184206 IC50 = 185 nM T23499 C7D8KR 18184228 IC50 = 119 nM T23499 C6YPB0 18184229 IC50 = 80 nM T23499 CEO31D 18184234 IC50 = 45 nM T23499 C4MK2X 18184249 IC50 = 2193 nM T23499 CP3IL6 18184256 IC50 = 724 nM T23499 COB38T 18617284 IC50 = 2000 nM T23499 CG1TS0 18617288 IC50 = 79 nM T23499 CBV58I 18617299 IC50 = 14000 nM T23499 C9PW8A 18617302 IC50 = 160 nM T23499 C2PJ4H 18617303 IC50 = 120 nM T23499 CI7W0J 18617314 IC50 = 13000 nM T23499 CO3F6N 18617318 IC50 = 40 nM T23499 CNFU26 18617322 IC50 = 71 nM T23499 CSP2T0 18617327 IC50 = 140 nM T23499 C58ZQH 18617333 IC50 = 72 nM T23499 CB9CL8 18617340 IC50 = 29 nM T23499 C0LCU8 18617344 IC50 = 19000 nM T23499 CD7H9C 18617345 IC50 = 62 nM T23499 CT8U7N 18617351 IC50 = 110 nM T23499 CBS6A9 18617354 IC50 = 550 nM T23499 CAP5D3 18617355 IC50 = 1400 nM T23499 C7VJ0E 18617363 IC50 = 2500 nM T23499 CE2NL8 18617366 IC50 = 3000 nM T23499 CC27DW 18617374 IC50 = 230 nM T23499 C8V6XS 18617377 IC50 = 44 nM T23499 C3JH0V 18617379 IC50 = 170 nM T23499 C57JVD 18617381 IC50 = 990 nM T23499 CBXP49 18617385 IC50 = 10000 nM T23499 CB42AR 18617389 IC50 = 240 nM T23499 CFL1W8 18617393 IC50 = 27 nM T23499 CL5EW6 18617394 IC50 = 53000 nM T23499 C6Q7CR 18617395 IC50 = 2700 nM T23499 C5OH8G 18617403 IC50 = 230 nM T23499 CP0TM2 18617407 IC50 = 3800 nM T23499 CFVX48 18630945 IC50 = 1.4 nM T23499 C72QST 18660520 Ki = 6.2 nM T23499 CLMZ12 18660521 Ki = 2.3 nM T23499 C7R1HU 18660522 Ki = 25 nM T23499 C2L4ID 18660523 Ki = 300 nM T23499 C92SQL 18704814 IC50 = 39.81 nM T23499 CUX27H 18704821 IC50 = 31.62 nM T23499 CQ35FJ 18738878 IC50 = 3.5 nM T23499 CC23YB 18738879 IC50 = 32 nM T23499 CVMZ19 18738880 IC50 = 30 nM T23499 C0L6JX 18738881 IC50 = 22 nM T23499 CZ8G6A 18738889 IC50 = 210 nM T23499 C82XBV 18738890 IC50 = 100 nM T23499 CW5JB8 18995986 IC50 = 170 nM T23499 CKJ26Q 18995988 IC50 = 4600 nM T23499 C89KDZ 18995989 IC50 = 620 nM T23499 CUL4T0 18995990 IC50 = 380 nM T23499 CZO82K 18995991 IC50 = 64 nM T23499 CZMR43 18995992 IC50 = 41 nM T23499 CSR67J 18995995 IC50 > 2500 nM T23499 C8CU9J 18995996 IC50 = 81 nM T23499 C24WKM 18995998 IC50 = 58 nM T23499 CIY7D1 18995999 IC50 = 84 nM T23499 CG4T2P 18996000 IC50 = 590 nM T23499 C41WAQ 19010490 IC50 = 700 nM T23499 C8CPZ7 19010493 IC50 = 38 nM T23499 CFK4N3 19010508 IC50 = 840 nM T23499 CGQL06 19085508 Ki = 220 nM T23499 CJ4W8X 19085510 Ki = 3.3 nM T23499 C6KS9O 19095644 IC50 = 800 nM T23499 C5YOI3 19347988 IC50 = 5900 nM T23499 CE49LB 19385674 IC50 = 11000 nM T23499 CAH21E 19432649 IC50 = 1500 nM T23499 CH9GX2 19432672 IC50 = 80 nM T23499 C6OW3M 19735343 IC50 = 18000 nM T23499 C69UIM 19735404 IC50 = 2000 nM T23499 C8FBX0 19934534 Ki = 33000 nM T23499 CO9WQ2 19934535 Ki = 80000 nM T23499 CC16NT 19934540 Ki = 109000 nM T23499 C8R7YA 19934544 Ki = 14000 nM T23499 CGEO10 19934546 Ki = 7000 nM T23499 C7YT0O 19934549 Ki = 41000 nM T23499 C3NT6Q 20747572 Ki = 700 nM T23499 CR28VH 20747573 Ki = 22 nM T23499 CL1CR3 20747574 Ki = 4 nM T23499 C5FZX8 20747575 Ki = 7 nM T23499 C38JIZ 21041249 IC50 = 4.3 nM T23499 CYNS68 21041264 IC50 = 0.3 nM T23499 C0EG5I 21041266 IC50 = 4.4 nM T23499 C9WM5T 21041267 IC50 = 1.7 nM T23499 C6R5QB 21041273 IC50 = 2.4 nM T23499 CSU45B 21041278 IC50 = 0.1 nM T23499 CM56UH 21041283 IC50 = 0.5 nM T23499 C50SCK 21041284 IC50 = 0.3 nM T23499 CTH8F6 21041288 IC50 = 2 nM T23499 C5JIK7 21041297 IC50 = 1.5 nM T23499 CIVT14 21041307 IC50 = 3.3 nM T23499 CA5U7Z 21041324 IC50 = 1.2 nM T23499 CQ63RK 21041370 IC50 = 1.4 nM T23499 C91PNA 21041372 IC50 = 1.4 nM T23499 CAK1Q0 21559921 IC50 > 25000 nM T23499 CGC23S 21559928 IC50 > 25000 nM T23499 C8QSU9 21979593 IC50 = 1.4 nM T23499 CB5KF0 21979601 IC50 = 6.9 nM T23499 CB7YS6 22009947 IC50 = 5.3 nM T23499 C6O5CM 22103385 Ki = 4 nM T23499 C4FDK6 22103537 Ki = 270 nM T23499 CQ2NK5 22103589 Ki = 44 nM T23499 C02YLT 22103743 Ki = 5.6 nM T23499 CLX1H5 22103787 Ki = 6.7 nM T23499 C60JDI 22103797 Ki = 19 nM T23499 CJ0UH7 22467219 IC50 = 34 nM T23499 C6G9YF 22467229 IC50 = 38 nM T23499 CSKR05 22467230 IC50 = 8.8 nM T23499 CVK24H 22467231 IC50 = 61 nM T23499 CRZI09 22467234 IC50 = 1.4 nM T23499 CN21KV 22467235 IC50 = 2.3 nM T23499 CASM08 22467237 IC50 = 1.7 nM T23499 C2B4MU 22467240 IC50 = 35 nM T23499 C21FKO 22467266 IC50 = 8.7 nM T23499 C1JMB2 22574645 Ki = 8 nM T23499 C8JZT4 22574723 Ki = 7 nM T23499 C0ZFH4 22574798 Ki = 20 nM T23499 CHF5V9 22616255 IC50 = 90000 nM T23499 CA1RM2 22616257 IC50 = 140 nM T23499 C0D9JA 22616258 IC50 = 15.6 nM T23499 CV3O7Y 22616262 IC50 = 110 nM T23499 CJTM39 22998396 IC50 = 603 nM T23499 CI8EP7 22998414 IC50 = 6140 nM T23499 CV17XE 22998438 IC50 = 680 nM T23499 CC4V5I 22998439 IC50 = 2520 nM T23499 C72NFC 22998446 IC50 = 36600 nM T23499 CR3HW0 22998447 IC50 = 1450 nM T23499 C15ZYN 22998456 IC50 = 104 nM T23499 CD91IN 22998508 IC50 = 315.5 nM T23499 CD6SZ3 23288645 IC50 > 100000 nM T23499 C3C4PE 23445219 IC50 = 1320 nM T23499 CIJ1C5 23445221 IC50 = 290 nM T23499 C68XCT 23445224 IC50 = 270 nM T23499 CA0G8O 23445227 IC50 = 299 nM T23499 C6E2OR 23445241 IC50 = 2710 nM T23499 C4J7YM 23445250 IC50 = 47.9 nM T23499 CTCP41 23445254 IC50 = 2603 nM T23499 CX95AD 23445256 IC50 = 205 nM T23499 CGN9I1 23445272 IC50 = 347 nM T23499 CEU2K7 23445284 IC50 = 217.5 nM T23499 CJ9U1W 23445285 IC50 = 159.6 nM T23499 C1QT2W 23445304 IC50 = 62 nM T23499 C2EB0A 23445313 IC50 = 54 nM T23499 CNJM59 23445317 IC50 = 1200 nM T23499 CG1P3S 23445325 IC50 = 148 nM T23499 C68HIG 23445333 IC50 = 91 nM T23499 CCMH86 23445336 IC50 = 58 nM T23499 C9I3JT 23445345 IC50 = 4120 nM T23499 C4AG5C 23445354 IC50 = 184 nM T23499 CT2F4G 23445355 IC50 = 0.04 nM T23499 C4T5MS 23445358 IC50 = 832 nM T23499 CCA74M 23445366 IC50 = 115 nM T23499 C4Z1GC 23445379 IC50 = 308 nM T23499 CN3G8K 23445388 IC50 = 819 nM T23499 CSP3J7 23445404 IC50 = 9.3 nM T23499 C5S0AP 23445408 IC50 = 82.3 nM T23499 CCJ37R 23445410 IC50 = 306 nM T23499 CGW8P2 23445412 IC50 = 650 nM T23499 C7B6HX 23445421 IC50 = 102 nM T23499 CZC52A 23445430 IC50 = 231 nM T23499 CYF1C9 23445438 IC50 = 237 nM T23499 C8AF2V 23445445 IC50 = 550 nM T23499 C5WR4F 23445457 IC50 = 62 nM T23499 CV1ER8 23445458 IC50 = 218 nM T23499 CNM0T8 23445468 IC50 = 65 nM T23499 C0VA4G 23445498 IC50 = 100.2 nM T23499 CIC27H 23445505 IC50 = 3220 nM T23499 C17QTN 23445506 IC50 = 1710 nM T23499 CV1TW8 23445507 IC50 = 1200 nM T23499 C4D0BK 23445516 IC50 = 182 nM T23499 C2G0WY 23445523 IC50 = 513 nM T23499 C0VE5Q 23445533 IC50 = 55 nM T23499 CIU74B 23445537 IC50 = 134 nM T23499 CAM4F5 23445538 IC50 = 346 nM T23499 C8S6HK 23445544 IC50 = 936 nM T23499 C64LFR 23445547 IC50 = 3390 nM T23499 CV6ZO3 23445562 IC50 = 4400 nM T23499 C1CUD7 23445593 IC50 = 106 nM T23499 CK28IV 23548251 IC50 = 4775 nM T23499 C7R6ZY 23548253 IC50 = 2.2 nM T23499 C6QBP1 23662235 Ki = 0.015 nM T23499 CZP9W1 23665178 IC50 = 7.4 nM T23499 CA50BD 23690609 IC50 = 0.38 nM T23499 CG74JF 23705748 IC50 = 10 nM T23499 CHQI17 23705749 IC50 = 0.98 nM T23499 C32JUQ 24997097 IC50 = 37.01 nM T23499 CW9D6N 25211074 IC50 = 0.11 nM T23499 C7LI1Q 42630531 IC50 = 13.5 nM T23499 C8TE1M 42630532 IC50 = 38.1 nM T23499 CW8MG1 42630654 IC50 = 24.4 nM T23499 CL63TM 42630655 IC50 = 1.44 nM T23499 C05NBA 44177614 IC50 = 373 nM T23499 CR8I5W 44211959 IC50 = 500 nM T23499 CS6L8E 44212539 IC50 = 6 nM T23499 CXWM12 44213540 Ki = 37 nM T23499 CHS1V8 44213651 IC50 = 900 nM T23499 C7KP1R 44213959 IC50 = 13000 nM T23499 CY6UZ1 44214320 IC50 = 14 nM T23499 CGP2D6 44215416 IC50 = 6 nM T23499 CU6GE5 44265871 Ki = 6.5 nM T23499 C6TNJ7 44266532 IC50 = 4100 nM T23499 C3B0YZ 44266537 IC50 = 2700 nM T23499 CQLH23 44266538 IC50 = 11000 nM T23499 CEN40G 44266540 IC50 = 1500 nM T23499 C3VGW6 44266542 IC50 = 800 nM T23499 CVJ34I 44266549 IC50 = 1500 nM T23499 CTBY61 44266552 IC50 = 80 nM T23499 CB8AT5 44266565 IC50 = 1100 nM T23499 C5L4PX 44266567 IC50 = 80 nM T23499 CQX4I8 44266568 IC50 = 2400 nM T23499 CD3L0E 44266575 IC50 = 43 nM T23499 CL6R1C 44266592 IC50 = 260 nM T23499 C4KI0U 44266594 IC50 = 60 nM T23499 C3JPQ4 44266595 IC50 = 1300 nM T23499 CPU56S 44266621 IC50 = 7400 nM T23499 C9FZ2P 44266628 IC50 = 5500 nM T23499 C7UH4R 44266629 IC50 = 2300 nM T23499 CT7VN2 44266640 IC50 = 240 nM T23499 CTP3M2 44266645 IC50 = 3500 nM T23499 CDI8R1 44266646 IC50 = 60 nM T23499 C6IW4B 44266649 IC50 = 10000 nM T23499 CN97HS 44266654 IC50 = 12000 nM T23499 CE8C3V 44266655 IC50 = 350 nM T23499 CQ0G4Y 44266850 IC50 = 0.78 nM T23499 C4T2NO 44266881 IC50 = 4.9 nM T23499 CNL7H5 44266886 IC50 = 1.1 nM T23499 C95YDQ 44266902 IC50 = 0.34 nM T23499 CC5IY6 44266940 IC50 = 49 nM T23499 C4K0DX 44267002 IC50 = 16000 nM T23499 CE8D3Z 44267860 Ki = 20 nM T23499 CVOS70 44267862 Ki = 15 nM T23499 CG7EO8 44267891 Ki = 105 nM T23499 CMRX95 44267893 Ki = 16 nM T23499 C53IRS 44270498 IC50 = 75 nM T23499 CB5YF6 44270522 IC50 = 600 nM T23499 CXM1K7 44270523 IC50 = 330 nM T23499 CV5SA1 44270524 IC50 = 1600 nM T23499 CG5ZR9 44270602 IC50 = 820 nM T23499 C0WCV2 44274885 Ki = 160 nM T23499 CJY0N4 44274960 Ki = 250 nM T23499 C8UH9L 44275660 Ki = 0.01 nM T23499 CC0B8Z 44277840 Ki = 0.01 nM T23499 CJ9Q2O 44278003 IC50 = 160 nM T23499 C9PSJ0 44278161 IC50 = 20000 nM T23499 C7OHT4 44278215 IC50 = 100 nM T23499 C0GRH9 44278270 IC50 = 23000 nM T23499 C8UGF0 44279126 IC50 = 7600 nM T23499 C8B5ID 44279127 IC50 = 47 nM T23499 C6BWO0 44279128 IC50 = 530 nM T23499 C2SQY1 44279129 IC50 = 48000 nM T23499 CZ5H9U 44279140 IC50 = 199.53 nM T23499 C29YIW 44279141 IC50 = 0.631 nM T23499 CQ90TU 44279172 IC50 = 3.981 nM T23499 C07WKA 44279173 IC50 = 39.81 nM T23499 CWI9G8 44279237 IC50 = 39.81 nM T23499 C2GJ3U 44279294 IC50 = 1 nM T23499 C08POS 44279295 IC50 = 2.512 nM T23499 CU2M7O 44279296 IC50 = 1.259 nM T23499 CJ51RL 44279303 IC50 = 1.585 nM T23499 CA7CE3 44279309 IC50 = 150 nM T23499 CFIK31 44279316 IC50 = 0.7943 nM T23499 CY7G4S 44279349 IC50 = 15000 nM T23499 CD19IQ 44279350 IC50 = 3900 nM T23499 CMK16B 44279351 IC50 = 5000 nM T23499 CS94JH 44279370 IC50 = 350 nM T23499 CJ5KZ3 44279371 IC50 = 26000 nM T23499 C0HE1T 44279383 IC50 = 290 nM T23499 C4M0NL 44279398 IC50 = 1 nM T23499 CIU3Q9 44279413 IC50 = 400 nM T23499 CZ0J7H 44279439 IC50 = 25000 nM T23499 C0N1IA 44279554 IC50 = 0.5012 nM T23499 CP3D7U 44279677 IC50 = 650 nM T23499 C04CFK 44283270 IC50 = 6100 nM T23499 C1Z9MO 44283471 IC50 = 16 nM T23499 C8PY9L 44284041 IC50 = 0.057 nM T23499 CR8I5H 44284115 IC50 = 0.041 nM T23499 CRTC24 44284183 IC50 = 0.86 nM T23499 C0R8DG 44284184 IC50 = 0.74 nM T23499 C8DOW0 44284196 IC50 = 0.41 nM T23499 CG38VX 44284199 IC50 = 0.8 nM T23499 CHR04C 44284236 IC50 = 0.022 nM T23499 CPDN49 44284238 IC50 = 0.031 nM T23499 C12RKH 44284266 IC50 = 0.027 nM T23499 C58KJR 44284284 IC50 = 8900 nM T23499 C16MGW 44284287 IC50 = 0.045 nM T23499 CB6IV3 44284288 IC50 = 0.014 nM T23499 CEJ9P3 44284292 IC50 = 0.014 nM T23499 CW2VK0 44284328 IC50 = 0.047 nM T23499 CQS3K4 44284329 IC50 = 0.11 nM T23499 CFSM06 44284381 IC50 = 0.22 nM T23499 C0YEI3 44284385 IC50 > 50000 nM T23499 CBP0H2 44284391 IC50 = 0.065 nM T23499 C02HIZ 44284405 IC50 = 0.011 nM T23499 C3PU2W 44284437 IC50 = 0.011 nM T23499 CJ04KH 44286764 Ki = 11222 nM T23499 C0UXK5 44291255 IC50 = 3 nM T23499 C8LI6J 44291575 IC50 = 3.4 nM T23499 CKON69 44291583 IC50 = 10.8 nM T23499 C20VYP 44291584 IC50 = 1430 nM T23499 C3QT4K 44291602 IC50 = 549 nM T23499 CC95RE 44291884 IC50 = 10 nM T23499 C24SGF 44291897 IC50 = 3.9 nM T23499 C0C5NJ 44293417 IC50 = 14 nM T23499 CQ67FH 44293526 IC50 = 68 nM T23499 C2AGE5 44293547 IC50 > 10000 nM T23499 CX4Q0F 44293631 IC50 = 58 nM T23499 C6OW4C 44293661 IC50 > 10000 nM T23499 CI71LD 44293681 IC50 > 10000 nM T23499 CPO24D 44293682 IC50 = 95 nM T23499 CKW14A 44293685 IC50 = 85 nM T23499 CQ3SJ6 44293702 IC50 > 10000 nM T23499 C3TIY5 44293716 IC50 = 3300 nM T23499 C7E6ZX 44293719 IC50 = 310 nM T23499 C9TPC5 44293720 IC50 = 6.1 nM T23499 C4KB5G 44293736 IC50 = 77 nM T23499 CNM5Z8 44293741 IC50 = 96 nM T23499 C7QP0V 44293754 IC50 = 31 nM T23499 C41MXT 44293761 IC50 = 22 nM T23499 C9J5CF 44293805 IC50 = 29 nM T23499 CMX3L8 44293813 IC50 = 330 nM T23499 C8S6BL 44293825 IC50 > 1000 nM T23499 C3JVX8 44293866 IC50 = 120 nM T23499 C6IRG7 44293868 IC50 = 96 nM T23499 CS60JA 44293907 IC50 > 10000 nM T23499 C9B7VD 44293915 IC50 = 1100 nM T23499 CL9WP4 44293927 IC50 = 66 nM T23499 C9SK1O 44293932 IC50 = 110 nM T23499 CZ6B8O 44302513 IC50 = 12.36 nM T23499 CSF3D1 44302615 IC50 = 0.11 nM T23499 CWL42G 44303033 Ki = 170 nM T23499 CS6JP9 44303148 Ki = 400 nM T23499 CS80KW 44304492 IC50 = 4 nM T23499 CU73DW 44307287 Ki = 160 nM T23499 CWSO92 44307412 Ki = 250 nM T23499 C6UL9Q 44309488 IC50 = 2500 nM T23499 CGO1R4 44310016 IC50 = 33 nM T23499 CC3ZE2 44311135 IC50 = 6 nM T23499 CDSL53 44311218 IC50 = 1900 nM T23499 CSLX12 44311225 IC50 = 1100 nM T23499 CQJI05 44311232 IC50 = 4 nM T23499 C9KM0C 44311233 IC50 = 4 nM T23499 CR0E5T 44311283 IC50 = 14 nM T23499 COLR05 44311284 IC50 = 7 nM T23499 CW3M6Y 44311285 IC50 = 9 nM T23499 CBM46T 44311288 IC50 = 880 nM T23499 C01CDF 44311321 IC50 = 900 nM T23499 CLRE28 44311345 IC50 = 3 nM T23499 CN7C4F 44311346 IC50 = 1 nM T23499 CR06YA 44311516 IC50 = 17 nM T23499 CNR47S 44311527 IC50 = 30 nM T23499 CVI91E 44311528 IC50 = 7 nM T23499 CPT62F 44311692 Ki = 0.89 nM T23499 CL5KJ1 44311698 Ki = 2300 nM T23499 C0GZL9 44311699 Ki = 250 nM T23499 CE5RU8 44311700 Ki = 54 nM T23499 C6COX5 44311701 Ki = 45 nM T23499 CC30ZG 44311726 Ki = 3.9 nM T23499 CB3G2V 44311727 Ki = 2.2 nM T23499 C9J6SX 44311728 Ki = 1.9 nM T23499 CIL3K7 44311763 Ki = 8 nM T23499 CUD78H 44311772 Ki = 5.2 nM T23499 CTCJ29 44311773 Ki = 5.5 nM T23499 C1YQW0 44311803 Ki = 6 nM T23499 CYV6P0 44311804 Ki = 2.9 nM T23499 C2ZN5I 44311805 Ki = 10 nM T23499 CEGV56 44311810 Ki = 850 nM T23499 C10LVB 44311838 Ki = 5.3 nM T23499 CD6AW7 44311849 Ki = 3.1 nM T23499 CF01CS 44311850 Ki = 5.4 nM T23499 C9B4XY 44311851 Ki = 130 nM T23499 CV1DH5 44311852 Ki = 87 nM T23499 C40EXJ 44311858 Ki = 9.1 nM T23499 CJD0Y3 44311873 Ki = 8.6 nM T23499 C45IUQ 44311915 Ki = 2.3 nM T23499 CXSC73 44311989 Ki = 6.9 nM T23499 CM4JA6 44312023 Ki = 27000 nM T23499 CB3YW0 44314173 IC50 = 8.6 nM T23499 CM2NJ4 44314579 IC50 = 2400 nM T23499 C80SJM 44314619 IC50 = 13 nM T23499 CMNS53 44314802 IC50 = 2.9 nM T23499 C7AS9N 44314904 IC50 = 3 nM T23499 C1LU5S 44315008 IC50 = 6.4 nM T23499 CY36NW 44316458 IC50 = 490 nM T23499 C39PCZ 44316515 IC50 = 470 nM T23499 C4NZK2 44316526 IC50 = 840 nM T23499 CYWQ80 44316527 IC50 = 270 nM T23499 C3B2EK 44316685 IC50 = 1000 nM T23499 COL70Q 44316686 IC50 = 980 nM T23499 CUG3R0 44316768 IC50 = 53 nM T23499 CV0FY7 44316831 IC50 = 270 nM T23499 CM0X9O 44316973 IC50 = 1800 nM T23499 CK8Z2M 44316983 IC50 = 1900 nM T23499 CNI1P7 44316993 IC50 = 1500 nM T23499 C65TIZ 44316994 IC50 = 720 nM T23499 CKY04J 44317005 IC50 = 430 nM T23499 C4ED2W 44317109 IC50 = 140 nM T23499 CSO8W9 44317215 IC50 = 4200 nM T23499 C39TVL 44320243 Ki = 224 nM T23499 CE06HD 44320537 Ki = 83000 nM T23499 C2ED3M 44320735 IC50 = 1800 nM T23499 C4PIJ8 44320779 IC50 = 8000 nM T23499 C6XZ9F 44320780 IC50 > 10000 nM T23499 CROU05 44320906 IC50 = 6700 nM T23499 CG1M6U 44320907 IC50 = 3600 nM T23499 C3USP1 44320908 IC50 > 10000 nM T23499 CRB52L 44321030 IC50 = 400 nM T23499 C59RKB 44321031 IC50 > 10000 nM T23499 CYEC03 44321032 IC50 = 8000 nM T23499 CS56NQ 44321033 IC50 = 9100 nM T23499 CTKV38 44321073 IC50 > 10000 nM T23499 CNH7R6 44321074 IC50 > 10000 nM T23499 C2M1KR 44321075 IC50 > 10000 nM T23499 CP29DA 44321080 IC50 > 10000 nM T23499 C4VT1P 44321081 IC50 = 1180 nM T23499 CCTK58 44321082 EC50 = 25 nM T23499 CTM7Z8 44321103 IC50 = 18400 nM T23499 C73YWI 44321104 IC50 > 10000 nM T23499 CNQU30 44321119 IC50 = 420 nM T23499 CSCV28 44321124 IC50 = 930 nM T23499 C5A1UD 44321125 IC50 > 100000 nM T23499 CKY10Z 44321131 IC50 = 14000 nM T23499 CGMA24 44321132 IC50 > 10000 nM T23499 C5TMZ2 44321226 IC50 = 200 nM T23499 CI7VO0 44322947 IC50 = 334 nM T23499 CU3VH5 44327347 IC50 = 3600 nM T23499 CZX9H8 44327348 IC50 = 2600 nM T23499 CNE6D9 44327437 IC50 = 13 nM T23499 CSD01Y 44327438 IC50 = 130 nM T23499 CV5YJ0 44327466 IC50 = 10000 nM T23499 C6ABP5 44327568 IC50 = 2000 nM T23499 CVOB31 44327585 IC50 = 6200 nM T23499 CF91QO 44327628 IC50 = 540 nM T23499 CU3HD9 44327629 IC50 = 36 nM T23499 C5M4ZA 44327656 IC50 = 250 nM T23499 C62PSA 44327659 IC50 = 230 nM T23499 CQCA89 44327660 IC50 = 1900 nM T23499 C3BLO7 44327778 IC50 = 4000 nM T23499 CNV45R 44327779 IC50 > 10000 nM T23499 C7XVA5 44327821 IC50 = 850 nM T23499 CJM4G3 44327853 IC50 = 2100 nM T23499 CR3X8K 44327867 IC50 = 11000 nM T23499 C93SIT 44327868 IC50 = 3200 nM T23499 CYG4E5 44327869 IC50 = 500 nM T23499 CBRK19 44327870 IC50 = 420 nM T23499 C9R8WV 44327875 IC50 > 10000 nM T23499 C3EH2T 44327876 IC50 = 320 nM T23499 CQL2D8 44327881 IC50 = 3500 nM T23499 CF69ID 44327889 IC50 > 10000 nM T23499 CF28EL 44327890 IC50 = 6300 nM T23499 C0N8PA 44327891 IC50 = 650 nM T23499 C0M1PO 44327892 IC50 = 17 nM T23499 CJI3F5 44327902 IC50 = 68 nM T23499 CLKA68 44327903 IC50 = 160 nM T23499 C69GCN 44327931 IC50 > 10000 nM T23499 CWGY59 44328018 IC50 = 380 nM T23499 CG6N2W 44328019 IC50 = 2600 nM T23499 C9NZT0 44328042 IC50 = 230 nM T23499 CQY25E 44328057 IC50 = 5000 nM T23499 CKD86E 44328060 IC50 = 140 nM T23499 C26WPT 44328073 IC50 > 10000 nM T23499 CBZ3U7 44328087 IC50 = 580 nM T23499 C4WS7B 44328089 IC50 = 21 nM T23499 CT9O6X 44328090 IC50 > 10000 nM T23499 CP67KV 44328091 IC50 = 450 nM T23499 C4FJ9U 44328092 IC50 = 35 nM T23499 CXA79S 44332345 IC50 > 25000 nM T23499 C8Z2AX 44332361 IC50 > 25000 nM T23499 CKYJ08 44332546 IC50 = 8700 nM T23499 COS3A7 44332577 IC50 = 1500 nM T23499 C1EC0A 44332578 IC50 = 5600 nM T23499 C76DUS 44332623 IC50 = 13000 nM T23499 CFO9I7 44332624 IC50 = 7900 nM T23499 CO8R3A 44332638 IC50 = 8200 nM T23499 CZ1AQ5 44332641 IC50 > 25000 nM T23499 C4OKR9 44332650 IC50 > 25000 nM T23499 C28FPG 44332656 IC50 > 25000 nM T23499 C6J3WT 44332735 IC50 = 0.4 nM T23499 CDC7Y9 44332745 IC50 > 25000 nM T23499 CTW54G 44332775 IC50 > 25000 nM T23499 C65INQ 44332776 IC50 > 25000 nM T23499 CO0J2A 44332777 IC50 > 25000 nM T23499 C4Q7DP 44332803 IC50 = 2800 nM T23499 CHL52J 44332807 IC50 = 57000 nM T23499 C7AGX8 44332823 IC50 > 25000 nM T23499 CSKC13 44332824 IC50 > 25000 nM T23499 CL7P8D 44332842 IC50 = 1 nM T23499 C1FCX4 44332856 IC50 > 25000 nM T23499 C5LV3A 44333055 IC50 > 25000 nM T23499 CGBP95 44333056 IC50 > 25000 nM T23499 CIE78D 44333366 Ki = 105 nM T23499 CBRP45 44333578 IC50 = 4.5 nM T23499 CKC04D 44333598 IC50 = 0.92 nM T23499 C2BM9V 44333721 IC50 = 0.51 nM T23499 CU74CY 44333867 IC50 = 5.7 nM T23499 CL8Q2W 44333887 IC50 = 7 nM T23499 C48LXP 44333889 IC50 = 8.2 nM T23499 CS3HR9 44333913 IC50 = 0.37 nM T23499 C6BH7M 44334053 IC50 = 15 nM T23499 CNBR86 44334065 IC50 = 1.6 nM T23499 C0QDY5 44334084 IC50 = 150 nM T23499 C3QKF4 44334097 IC50 = 0.55 nM T23499 C7VSP8 44334128 IC50 = 0.2 nM T23499 CXR8T9 44334129 IC50 = 1.9 nM T23499 CK0C1Y 44334130 IC50 = 2.2 nM T23499 C0BX8D 44334145 IC50 = 3.2 nM T23499 C1I5CL 44334146 IC50 = 0.12 nM T23499 C4BJ7O 44334150 IC50 = 0.32 nM T23499 C1A2MU 44339655 IC50 = 0.29 nM T23499 C8N7UJ 44339756 Ki = 0.43 nM T23499 C2H4FY 44340049 IC50 = 1 nM T23499 CM37XP 44357035 IC50 = 590 nM T23499 CHE24D 44357132 IC50 = 3.4 nM T23499 C9U6VC 44357174 IC50 = 8.3 nM T23499 CITF21 44357212 IC50 = 30 nM T23499 CY69NR 44357391 IC50 = 1.2 nM T23499 CH06JK 44364480 IC50 = 930 nM T23499 C07DXP 44364522 IC50 = 650 nM T23499 CUXG74 44365561 Ki = 38 nM T23499 C3W9KH 44365878 Ki = 3800 nM T23499 CR2SD4 44365953 IC50 < 800 nM T23499 CMTX03 44365954 IC50 = 30 nM T23499 CGVT83 44366010 IC50 = 15 nM T23499 CEO85C 44366033 IC50 = 130 nM T23499 C3G9XR 44366059 IC50 = 400 nM T23499 CZJ6C0 44368812 IC50 > 10000 nM T23499 C0F8EI 44371612 IC50 > 25000 nM T23499 CP3T7Z 44371671 IC50 = 8100 nM T23499 C2T7JL 44382933 IC50 = 140 nM T23499 CX20AK 44382975 IC50 = 1100 nM T23499 CH1JD4 44382976 IC50 = 1320 nM T23499 CFB19N 44383187 IC50 = 420 nM T23499 CG17CU 44383188 IC50 > 3500 nM T23499 CXAL80 44383189 IC50 = 295 nM T23499 CS15AY 44383241 IC50 = 220 nM T23499 C0Y1FZ 44383330 IC50 = 730 nM T23499 CV5B9Z 44383535 IC50 = 8200 nM T23499 CZ07MY 44383536 IC50 = 50000 nM T23499 CTR86P 44383537 IC50 = 62000 nM T23499 CF5J9H 44383572 IC50 > 3500 nM T23499 CHM06G 44383573 IC50 > 3500 nM T23499 CA7BX1 44383592 IC50 = 135000 nM T23499 CCM25J 44383602 IC50 = 8 nM T23499 CB2H4W 44383742 IC50 = 180 nM T23499 CWC95L 44383753 IC50 = 44 nM T23499 CYM1J5 44383754 IC50 = 166 nM T23499 CC4EQ1 44384177 IC50 = 129 nM T23499 C5CK8M 44384557 IC50 = 339 nM T23499 CS57OV 44384610 IC50 = 2770 nM T23499 CX4B1W 44384611 IC50 = 84 nM T23499 CSY82J 44384651 IC50 = 79 nM T23499 CK9W5F 44384652 IC50 = 73 nM T23499 C4M7YA 44384656 IC50 = 141 nM T23499 CQXM63 44384715 IC50 = 85 nM T23499 C1N3SA 44384723 IC50 = 582 nM T23499 CWQ32E 44384757 IC50 = 81 nM T23499 CDM4X3 44384766 IC50 = 96 nM T23499 C9ST7O 44384826 IC50 = 239 nM T23499 C3ZO9F 44384852 IC50 = 176 nM T23499 C3IH2N 44384966 IC50 = 186 nM T23499 CSJ42C 44385008 IC50 = 38 nM T23499 CUF05M 44385127 IC50 = 72 nM T23499 CJ02XC 44385162 IC50 = 11 nM T23499 C43ADQ 44385412 IC50 = 2190 nM T23499 CSP1A8 44385522 IC50 = 487 nM T23499 C35IMP 44385523 IC50 = 4900 nM T23499 C26DIF 44385576 IC50 = 121 nM T23499 C2E3SP 44385586 IC50 = 125 nM T23499 C4B8VR 44385792 IC50 = 1850 nM T23499 CG94RA 44385805 IC50 = 339 nM T23499 CYV8Q4 44386002 IC50 = 94 nM T23499 C6OYN9 44386069 IC50 = 8390 nM T23499 CE42KT 44386161 IC50 = 59 nM T23499 CADI16 44386162 IC50 = 165 nM T23499 CI87SP 44386163 IC50 = 1320 nM T23499 C3X1MN 44386169 IC50 = 0.4 nM T23499 CK7XM9 44387128 IC50 = 1700 nM T23499 CW4SK9 44387533 Ki = 81 nM T23499 CI8HL6 44404967 IC50 = 24 nM T23499 C0GO9C 44439102 IC50 = 1 nM T23499 CIS54Q 44439103 IC50 = 1.6 nM T23499 C97JIW 44439105 IC50 = 44.9 nM T23499 CE6RC7 44439106 IC50 = 8 nM T23499 CH7WG4 44439108 IC50 = 7.7 nM T23499 C3E1GM 44439111 IC50 = 4.6 nM T23499 C42LOW 44439114 IC50 = 21.6 nM T23499 CD4NM1 44458399 IC50 = 19 nM T23499 C8LEA4 44458597 IC50 = 3.1 nM T23499 CBUI18 44458604 IC50 = 6.5 nM T23499 CR69LH 44458650 IC50 = 5 nM T23499 C5BEX8 44458669 IC50 = 5.2 nM T23499 CV0S2K 44458670 IC50 = 2.8 nM T23499 CER1W7 44458999 IC50 = 7.5 nM T23499 CAJY18 44459247 IC50 = 72 nM T23499 CPT5A8 44459272 IC50 = 12 nM T23499 CVHR80 44459299 IC50 = 31 nM T23499 C4DL5C 44469677 IC50 > 10000 nM T23499 C37FQS 52943105 IC50 = 6.6 nM T23499 CER61Y 52943235 IC50 = 610 nM T23499 C05KUJ 52944083 IC50 = 9.9 nM T23499 C4YK3X 52944276 IC50 = 7.4 nM T23499 C68GJL 52949155 IC50 = 6.3 nM T23499 CMLQ42 52949197 IC50 = 115.9 nM T23499 CD4GT1 52950137 IC50 = 284.5 nM T23499 CPD2R7 54580805 IC50 = 60 nM T23499 C02NYX 56657875 IC50 = 260 nM T23499 CBNG90 56661220 IC50 = 13000 nM T23499 C2E6NA 56668088 IC50 = 14 nM T23499 CH6KE2 56668268 IC50 = 200 nM T23499 CI4B0R 56668269 IC50 = 700 nM T23499 C95DPK 56671553 IC50 = 30000 nM T23499 C5FP8A 56671554 IC50 > 25000 nM T23499 CW4R9X 56671734 IC50 = 250 nM T23499 CWP38Q 56674998 IC50 = 1800 nM T23499 C3KS9C 56678451 IC50 = 4500 nM T23499 CN4V1M 56678452 IC50 = 880 nM T23499 C0BU9Y 56679082 IC50 = 1 nM T23499 C2X1UN 56681797 IC50 = 2700 nM T23499 CR5A2Y 56681798 IC50 = 260 nM T23499 CQ35GN 56681799 IC50 = 3200 nM T23499 C8TSX9 58688005 IC50 = 0.7 nM T23499 CE97RP 58688006 IC50 = 0.3 nM T23499 C0IP5B 58688008 IC50 = 1.3 nM T23499 CY2NO8 66875612 IC50 = 1500 nM T23499 CU3B7D 67952994 IC50 = 1.6 nM T23499 C7ATS0 68169760 IC50 > 100000 nM T23499 CVO35E 70240112 IC50 = 33 nM T23499 C7CO8B 70684239 IC50 = 9.3 nM T23499 C7OTX0 70684240 IC50 = 11 nM T23499 C82TCO 70686380 IC50 = 99 nM T23499 CWK4N9 70686381 IC50 = 39 nM T23499 C6SLW4 70686382 IC50 = 9.8 nM T23499 CBXG08 70690542 IC50 = 10 nM T23499 C8XA7W 70692693 IC50 = 22 nM T23499 C3QC5F 70694736 IC50 = 75 nM T23499 CDJU89 70694737 IC50 = 8.9 nM T23499 CY9IA0 70694738 IC50 = 9.6 nM T23499 CL3ZU8 70696780 IC50 = 9.8 nM T23499 CH30FG 70696781 IC50 = 10 nM T23499 C0VJ2M 71449713 IC50 = 1.1 nM T23499 C49KEX 71451525 IC50 = 4.3 nM T23499 C7VJ0W 71451526 IC50 = 2.8 nM T23499 CR74NM 71451527 IC50 = 7.7 nM T23499 C1GA0F 71451528 IC50 = 4.3 nM T23499 CVA24Y 71451529 IC50 = 3.8 nM T23499 C2QI7H 71453356 IC50 = 1.9 nM T23499 CS79DP 71453357 IC50 = 1.5 nM T23499 CRD7T6 71455060 IC50 = 2.8 nM T23499 C9JZM4 71455061 IC50 = 739 nM T23499 CKL51C 71455062 IC50 = 3 nM T23499 CL4T8W 71455063 IC50 = 1.7 nM T23499 C4Q6LJ 71455064 IC50 = 7 nM T23499 CL76UZ 71455065 IC50 = 3.4 nM T23499 CB0EI6 71455139 IC50 = 6.8 nM T23499 CUV4P7 71455140 IC50 = 3.6 nM T23499 CYB60E 71456862 IC50 = 10.4 nM T23499 C7N3KS 71456863 IC50 = 1.9 nM T23499 C7LMX1 71456864 IC50 = 9.9 nM T23499 C3Q6IB 71456865 IC50 = 40 nM T23499 C4XE8T 71456935 IC50 > 100 nM T23499 CP5OM0 71458717 IC50 = 4534 nM T23499 C5ZC7W 71458718 IC50 = 17.8 nM T23499 CX2Q1M 71458719 IC50 = 1.1 nM T23499 CQ1C8Y 71458720 IC50 = 73 nM T23499 CJ0ZG5 71458721 IC50 = 14 nM T23499 C4H9GW 71460535 IC50 = 6.7 nM T23499 C3ZVU9 71460536 IC50 = 113 nM T23499 C07SOZ 71460537 IC50 = 187 nM T23499 CYS3W0 71460621 IC50 = 1 nM T23499 CA39BC 71462245 IC50 = 0.4 nM T23499 CX7C4B 71462246 IC50 = 7.9 nM T23499 CN3Z1G 71462247 IC50 = 2.1 nM T23499 CXG1J8 71462248 IC50 = 6.9 nM T23499 COUE65 71462320 IC50 = 0.7 nM T23499 CJCM28 71462321 IC50 = 2.3 nM T23499 CA78CN 71462322 IC50 = 0.8 nM T23499 CHX9P8 71719083 IC50 = 6200 nM T23499 CP2QW7 71719097 IC50 = 0.288 nM T23499 CWH6T3 72548703 IC50 = 0.023 nM T23499 CIY23Q 73345435 EC50 = 13 nM T23499 CQA8J6 73345452 IC50 = 5000 nM T23499 C5GF1A 73345478 IC50 = 18 nM T23499 CCP7Y5 73348424 IC50 > 50000 nM T23499 CAK0P5 73348425 IC50 = 30 nM T23499 CV41YQ 73348480 IC50 = 7100 nM T23499 CR3KM1 73348481 IC50 = 2200 nM T23499 CBY20F 73350002 IC50 = 3200 nM T23499 CM1HV9 73350041 EC50 = 2100 nM T23499 C25JCS 73350066 IC50 > 1000 nM T23499 C7SC3B 73351511 IC50 > 50000 nM T23499 C0R5BG 73352983 IC50 > 50000 nM T23499 C8R6GM 73354330 IC50 = 3000 nM T23499 CT6GP8 73354491 IC50 = 24000 nM T23499 C6NU5S 73354540 IC50 > 10000 nM T23499 CVR30I 73354541 IC50 > 10000 nM T23499 C1Q6RY 73356095 IC50 = 750 nM T23499 CD06SE 76308472 IC50 = 11 nM T23499 CVD37X 76312118 Ki = 2.2 nM T23499 CS4AO6 76319370 IC50 = 18 nM T23499 CVN3I8 76326542 IC50 = 560 nM T23499 C2G5FV 76330201 IC50 = 46 nM T23499 CEWB01 90663476 IC50 = 1300 nM T23499 CWY29O 90766557 IC50 = 2.2 nM T23499 CLI6Y5 101039204 IC50 = 7.3 nM T23499 CD6BY7 122194934 IC50 = 130 nM T23499 C5RKC4 122194935 IC50 = 112 nM T23499 CB0QI8 127026027 IC50 = 13000 nM T23499 CU0J4F 127026040 IC50 = 7100 nM T23499 C9QA0N 127026041 IC50 > 20000 nM T23499 C63KTY 127026042 IC50 = 9100 nM T23499 C8X0UC 127026043 IC50 = 165 nM T23499 CXN21Q 127026058 IC50 = 886 nM T23499 C4PWU0 127026336 IC50 > 20000 nM T23499 CFY04E 127026337 IC50 > 20000 nM T23499 C5YIM7 127026338 IC50 = 11000 nM T23499 C04OWP 127028595 IC50 > 20000 nM T23499 CSO5F2 127028617 IC50 > 20000 nM T23499 C1OFQ0 127028618 IC50 > 20000 nM T23499 C9OW0V 127028619 IC50 > 20000 nM T23499 CKY51I 127028620 IC50 > 20000 nM T23499 CVKG08 127028930 IC50 = 14000 nM T23499 CHP7W8 127029201 IC50 = 10000 nM T23499 CWSI52 127029202 IC50 = 126 nM T23499 CH5B3Y 127029203 IC50 = 7000 nM T23499 CS10YM 127029204 IC50 > 20000 nM T23499 C5UE4D 127034756 IC50 = 262 nM T23499 CWH4T7 127034757 IC50 = 56000 nM T23499 C5E4BU 127034758 IC50 = 24 nM T23499 CGVR16 127034901 IC50 = 1400 nM T23499 CT31NI 127034916 IC50 = 5800 nM T23499 CPL08Z 127034917 IC50 = 5500 nM T23499 CU39OI 127034918 IC50 = 35000 nM T23499 C64HFO 127034919 IC50 = 277 nM T23499 CZ61LK 127034966 EC50 > 5011.87 nM T23499 CA0SN5 127034967 EC50 > 5011.87 nM T23499 C5XM0K 127035067 IC50 = 1800 nM T23499 C1QJ0V 127035068 IC50 = 27000 nM T23499 CBC74Y 127035069 IC50 = 137 nM T23499 C67FNJ 127035070 IC50 = 10 nM T23499 CL01XK 127035082 IC50 = 898 nM T23499 CP6T3J 127035083 IC50 = 388 nM T23499 CJHG08 127035084 IC50 = 28000 nM T23499 CLJ94G 127035085 IC50 = 956 nM T23499 CRN65G 127035219 IC50 = 310 nM T23499 CE07IC 127035379 IC50 = 24000 nM T23499 C6DU4R 127035380 IC50 = 200000 nM T23499 C3XWN4 127035410 IC50 = 15 nM T23499 CA9FD3 127035544 IC50 = 3000 nM T23499 CF6X3E 127035545 IC50 = 55000 nM T23499 C5ED6S 127035757 IC50 = 11 nM T23499 CZN92T 127036865 IC50 = 10 nM T23499 C0KJO7 127036866 IC50 = 7200 nM T23499 C19VDE 127036867 IC50 = 625 nM T23499 C24HFS 127036868 IC50 > 20000 nM T23499 CPQB01 127037496 IC50 = 314 nM T23499 CEQS03 127037497 IC50 = 140000 nM T23499 CKUH43 134136255 IC50 = 75.4 nM T23499 C5G2PJ 134139749 IC50 = 693000 nM T23499 CC1N3A 134157696 IC50 = 0.67 nM T23499 C1GY2T 135156251 EC50 > 10000 nM T23499 C1LD6M 135415889 IC50 = 13 nM T23499 C8MXL7 135512539 IC50 = 22 nM T23499 CE1PR8 135870740 IC50 = 133000 nM T23499 C7O6VE 135884434 IC50 = 66 nM T23499 CN3ZE2 137633242 IC50 = 17.1 nM T23499 C23ACU 137633653 IC50 = 279.1 nM T23499 C9IRL3 137637038 IC50 = 1.2 nM T23499 CX0YV5 137638953 IC50 = 78.4 nM T23499 C7IM5Q 137639474 IC50 = 873 nM T23499 CDE50H 137642741 IC50 = 7.1 nM T23499 C81EDX 137643691 IC50 = 342 nM T23499 CA60GK 137647152 IC50 = 6.2 nM T23499 CW34UP 137649592 IC50 = 0.8 nM T23499 CQ8Y5V 137649809 IC50 = 1024 nM T23499 C09IFA 137652304 IC50 = 364.5 nM T23499 C1WG3B 137655285 IC50 = 373 nM T23499 CRT9I5 137655525 IC50 = 29.2 nM T23499 CD6W2K 137661460 IC50 = 48.2 nM T23499 C1MI4T 155511294 IC50 = 29 nM T23499 C49YIT 155517241 IC50 = 9.4 nM T23499 CD6GO2 155519245 IC50 = 35 nM T23499 C0YXP4 155519384 IC50 = 1 nM T23499 CGBM57 155535325 IC50 = 1300 nM T23499 CO8N9V 155542285 IC50 = 1.4 nM T23499 CZN9I0 155544917 IC50 = 0.5 nM T23499 CW6FD5 155551580 IC50 = 1 nM T23499 CF6T1B 155560343 IC50 = 1300 nM T23499 CJB9O1 155562688 IC50 = 15.4 nM T23499 CPEX85 155563100 IC50 = 2 nM T23499 CGH80Y 155564169 IC50 = 3 nM T23499 D00RGL 44371672 IC50 = 2400 nM T23499 D05ZUX 44207909 Ki >= 1000 nM T23499 D06OSN 44371614 IC50 = 9500 nM T23499 D07OMS 9960931 IC50 = 0.35 nM T23499 D0F8BZ 44371670 IC50 = 1900 nM T23499 D0FF6S 16038374 IC50 > 10000 nM T23499 D0G5UD 5312146 IC50 = 6800 nM T23499 D0M2TB 44368903 IC50 = 3800 nM T23499 D0NI1W 44368904 IC50 = 2600 nM T23499 D0T2RY 9948320 Ki >= 1000 nM T23499 D0W4UX 9908909 Ki = 4.7 nM T23499 D0X1XM 9893800 Ki = 2.15 nM T23499 D0X1ZC 9848710 Ki = 11000 nM T23499 D0Y1HN 5310991 IC50 = 8200 nM T23499 D0Y8UY 44371613 IC50 = 250 nM T38301 D0DT1R 9571836 IC50 = 185 nM T38301 CM3YC1 9555629 IC50 = 1000 nM T38301 C2V6ER 9571641 IC50 = 11000 nM T38301 CTYX93 10219945 IC50 = 1300 nM T38301 CXRW26 10513282 IC50 = 1000 nM T38301 C83NJC 10514912 IC50 = 2500 nM T38301 C6GO4F 10561865 IC50 = 1400 nM T38301 C7BKA4 10585847 IC50 = 1400 nM T38301 CC7KM5 10679937 IC50 = 2500 nM T38301 CU67EV 10681264 IC50 = 1700 nM T38301 CU15XV 10798500 IC50 = 9000 nM T38301 CK5GD4 44320830 IC50 = 820 nM T38301 C8ITE5 44320846 IC50 = 2700 nM T38301 C45IDJ 135458654 IC50 = 123000 nM T15439 D0G2XE 6918468 IC50 = 15.85 nM T15439 CU96IB 131577 Ki = 150000 nM T15439 CVJ46C 223995 IC50 > 100 ug.mL-1 T15439 C0LQG3 234070 IC50 > 100 ug.mL-1 T15439 CU3I9S 234079 IC50 > 100 ug.mL-1 T15439 CQ23YV 235632 IC50 > 60000 nM T15439 CQX4M9 265219 IC50 = 200 nM T15439 C7REB9 408239 IC50 > 50 ug.mL-1 T15439 CQJP09 1250946 EC50 > 60000 nM T15439 C03YNW 1351023 IC50 = 14600 nM T15439 C84SMK 1379975 IC50 = 8700 nM T15439 C39LPI 3196682 IC50 = 125.89 nM T15439 COT07B 3453336 IC50 = 59 nM T15439 C7MGQ3 5773323 IC50 = 12 ug.mL-1 T15439 CJ20TS 5909556 IC50 = 30 ug.mL-1 T15439 C2V4XW 9989013 EC50 = 48000 nM T15439 C9DA2N 10010954 IC50 = 490 nM T15439 CEM2F0 10011515 EC50 = 15800 nM T15439 CKI8Q7 10011643 EC50 = 2500 nM T15439 CR5SZ2 10057217 EC50 = 1200 nM T15439 CQ5IL1 10102925 EC50 = 4000 nM T15439 CXM30U 10260801 EC50 = 224000 nM T15439 C2L1OB 10328378 IC50 = 1995.26 nM T15439 CJ8L9B 10351296 EC50 = 300 nM T15439 C3J7VK 10351393 EC50 = 2100 nM T15439 CA17CG 10374110 EC50 = 5600 nM T15439 CMN41C 10374115 Ki = 390 nM T15439 C48BDO 10396578 EC50 = 4000 nM T15439 CM2C6S 10418298 IC50 = 360 nM T15439 CJFK61 10418799 EC50 = 215000 nM T15439 C3RMH6 10418817 EC50 = 19500 nM T15439 C0V2GR 10418881 EC50 = 22000 nM T15439 CUT40G 10441364 EC50 = 50000 nM T15439 CX0LR4 10441383 EC50 = 5000 nM T15439 CF3EV2 10463109 IC50 = 55000 nM T15439 CSO5E8 10464003 EC50 = 2300 nM T15439 CW8D9N 10464012 EC50 = 70000 nM T15439 C3OD5Q 10464120 EC50 = 500000 nM T15439 CRK13Y 10486513 IC50 = 4700 nM T15439 C7XFQ8 10510226 IC50 = 2600 nM T15439 C3MW1N 10557548 IC50 = 144000 nM T15439 CO7FW9 10557793 IC50 = 2951.21 nM T15439 CFY13C 10616508 IC50 = 2000 nM T15439 C0VUX7 10629679 IC50 = 5888.44 nM T15439 CP6KR5 10653515 IC50 = 51000 nM T15439 C1ONR5 10724409 IC50 = 700 nM T15439 CM7AT6 10724498 IC50 > 42657.95 nM T15439 C29SYI 10795799 IC50 = 12 nM T15439 CWA0K3 10796341 IC50 = 4570.88 nM T15439 CE3C2X 10819181 IC50 < 1000000 nM T15439 C6XU3O 10819260 IC50 = 9000 nM T15439 C5LQT4 10819534 IC50 = 500 nM T15439 CRA0F6 10843359 IC50 = 1949.84 nM T15439 CW1S3T 11766790 EC50 = 2000 nM T15439 C1OIT7 11803878 IC50 = 3548.13 nM T15439 CFUP74 11857314 IC50 = 90 nM T15439 C9T6HG 12253728 IC50 > 100000 nM T15439 CI0W3Z 12253756 IC50 = 30000 nM T15439 CCK8Z0 12473171 EC50 > 60000 nM T15439 C51CXK 14588192 IC50 = 1.7 ug.mL-1 T15439 C4NZ3E 15133383 IC50 = 2 ug.mL-1 T15439 COIX70 15133384 IC50 = 18 ug.mL-1 T15439 C2PY5T 15133385 IC50 > 50 ug.mL-1 T15439 C68FSN 15133387 IC50 > 100 ug.mL-1 T15439 CDXI20 15133388 IC50 > 50 ug.mL-1 T15439 C4UK1G 15133390 IC50 = 9 ug.mL-1 T15439 C9YG1I 15133392 IC50 > 50 ug.mL-1 T15439 CCB82L 15133393 IC50 > 100 ug.mL-1 T15439 C49TDH 15133396 IC50 > 100 ug.mL-1 T15439 CONB25 15133397 IC50 > 50 ug.mL-1 T15439 CM48AT 15133398 IC50 > 100 ug.mL-1 T15439 CLR8T7 15133399 IC50 = 8 ug.mL-1 T15439 CFBH58 15133400 IC50 = 30 ug.mL-1 T15439 C4ZHX7 15133401 IC50 = 30 ug.mL-1 T15439 C34QHN 15133402 IC50 = 4 ug.mL-1 T15439 CY6BQ4 15133403 IC50 = 7 ug.mL-1 T15439 C1RS9Y 15133405 IC50 > 100 ug.mL-1 T15439 CU54OK 15133406 IC50 > 100 ug.mL-1 T15439 C7NZE4 15133407 IC50 > 100 ug.mL-1 T15439 C8I5AS 15725946 Ki = 210000 nM T15439 C5PIR8 15725947 Ki = 25000 nM T15439 CGV6N1 15725948 Ki = 10000 nM T15439 CCF07N 15725949 Ki = 750000 nM T15439 CQJB30 15725952 Ki = 2900 nM T15439 CI9T5B 15725956 Ki = 2000 nM T15439 CK37JY 15725957 Ki = 1600 nM T15439 CW9YH0 15725958 Ki = 5300 nM T15439 C2Y3PS 17615045 IC50 = 44500 nM T15439 C1ZIJ0 24894075 IC50 = 7 nM T15439 CHR1V9 24970311 IC50 = 1 nM T15439 CLBN94 25010731 Ki = 8.9 nM T15439 CBJ5U6 25108851 IC50 = 51 nM T15439 CI0P1S 25109118 IC50 = 18 nM T15439 CY4IA6 25109473 IC50 = 26 nM T15439 CMF20W 25109614 IC50 = 25 nM T15439 C2QVM4 25109748 IC50 = 22 nM T15439 C9P8SK 25110775 IC50 = 125 nM T15439 C3Y7OS 25110776 IC50 = 90 nM T15439 CC0D4T 25191127 IC50 = 3200 nM T15439 CGO76M 25191129 IC50 = 3500 nM T15439 CN07LF 25191131 Ki = 3700 nM T15439 CH67ZI 25191132 IC50 = 4900 nM T15439 CDJY09 25191261 IC50 = 2600 nM T15439 CLTQ86 25191262 IC50 = 5000 nM T15439 C7ITF9 25191265 Ki = 370 nM T15439 C93JHW 25191266 IC50 = 6200 nM T15439 C6V1YK 25191388 Ki = 680 nM T15439 CG0WP7 25191514 IC50 = 6200 nM T15439 C28CUR 25191639 IC50 = 22 nM T15439 CCB8K5 25191640 IC50 = 26 nM T15439 C1FUH4 25191762 Ki = 21 nM T15439 C2XA8H 25191763 IC50 = 37 nM T15439 CV0HO8 25191764 IC50 = 53 nM T15439 CKR41V 25191765 IC50 = 67 nM T15439 C6A9NV 25191766 Ki = 13 nM T15439 CK2Z4S 25191896 IC50 = 82 nM T15439 C42QJX 25191897 Ki = 10 nM T15439 C9AUZ1 25191898 IC50 = 110 nM T15439 C5UC2L 25191899 Ki = 180 nM T15439 C3N6MS 25191900 IC50 = 120 nM T15439 CRJ5S2 25191901 IC50 = 130 nM T15439 CR01FX 25192049 Ki = 7.3 nM T15439 CDY74P 25192050 IC50 = 170 nM T15439 CB5DG7 25192196 IC50 = 180 nM T15439 CI1YP8 25192198 IC50 = 220 nM T15439 CUG5S4 25192200 Ki = 9.7 nM T15439 CE1FC6 25192335 IC50 = 270 nM T15439 C2DB6J 25192336 IC50 = 290 nM T15439 C57AGT 25192337 IC50 = 340 nM T15439 CR42YT 25192338 IC50 = 350 nM T15439 CD4J3C 25192339 Ki = 35 nM T15439 CUM4B7 25192488 IC50 = 410 nM T15439 CYS9R5 25192489 IC50 = 420 nM T15439 C6YI9W 25192490 IC50 = 430 nM T15439 C0HR8P 25192491 IC50 = 530 nM T15439 C2J9GL 25192493 IC50 = 560 nM T15439 CR0DC8 25192633 Ki = 86 nM T15439 CVHX47 25192634 IC50 = 690 nM T15439 CM3A6J 25192635 IC50 = 730 nM T15439 CM60NU 25192636 IC50 = 790 nM T15439 CJ3N7G 25192638 IC50 = 840 nM T15439 CATD54 25192764 IC50 = 880 nM T15439 CNU76Z 25192765 IC50 = 910 nM T15439 CCG2W3 25192766 IC50 = 950 nM T15439 C9T0DF 25192769 IC50 = 1400 nM T15439 C8ZQI3 25192896 IC50 = 1400 nM T15439 C3TG7E 25192897 IC50 = 1500 nM T15439 C1WAL2 25192898 IC50 = 1500 nM T15439 CAW5M1 25192901 IC50 = 1700 nM T15439 C25YCL 25193028 IC50 = 1700 nM T15439 CV04ES 25193029 Ki = 1200 nM T15439 C8SUH0 25193031 Ki = 180 nM T15439 C5TNI1 25193057 IC50 = 22 nM T15439 C8Q7VT 25193171 IC50 = 2400 nM T15439 CN24JP 25193172 IC50 = 2400 nM T15439 C2IP0H 25193174 IC50 = 2500 nM T15439 CB8ZC4 25193175 IC50 = 2600 nM T15439 C2L8UV 44301802 IC50 = 3090.3 nM T15439 CJ3R4O 44301857 IC50 > 16982.44 nM T15439 CIQ6K0 44301938 IC50 = 3200 nM T15439 CA96CM 44301960 IC50 = 16000 nM T15439 C6SI5F 44301966 IC50 = 41000 nM T15439 CC28KW 44301970 IC50 > 56.23 nM T15439 CWQG56 44301971 IC50 = 9500 nM T15439 CUT45G 44301983 IC50 > 269.15 nM T15439 C9VEY4 44301984 IC50 = 10000 nM T15439 CU58SH 44301986 IC50 = 300 nM T15439 CQ4N1X 44302015 IC50 = 3800 nM T15439 C56WNL 44302230 IC50 = 300 nM T15439 C4KS0O 44302231 IC50 = 8100 nM T15439 C2YPH6 44305324 Ki = 300000 nM T15439 CI0J4B 44305325 EC50 = 1.3 nM T15439 CO52KR 44305625 Ki = 100000 nM T15439 C5HD0K 44308822 IC50 = 4000 nM T15439 CI89BA 44342908 IC50 = 1800 nM T15439 CY5QI1 44347020 EC50 = 500000 nM T15439 CLB4Y1 44353001 Ki = 2100 nM T15439 C9Q5PJ 44353002 Ki = 260 nM T15439 CT89UX 44353003 Ki = 220 nM T15439 C4VP3O 44353014 Ki = 810 nM T15439 CFG6T2 44353020 Ki = 4400 nM T15439 C2BVM0 44353031 Ki = 36000 nM T15439 C7WVA2 44353032 Ki = 31000 nM T15439 CPJH61 44353033 Ki = 13000 nM T15439 CGCD74 44353083 Ki = 79000 nM T15439 C21JOP 44353179 Ki = 20000 nM T15439 C79ULO 44353181 Ki = 180000 nM T15439 CPJE52 44383008 IC50 = 8000 nM T15439 C4LIR7 44383043 IC50 = 50000 nM T15439 CE2F7V 44383126 IC50 = 4000 nM T15439 CY59VJ 44383127 IC50 = 6000 nM T15439 C17BQM 44383144 IC50 = 25000 nM T15439 CS92WK 44383275 IC50 = 4000 nM T15439 C1CM4J 44383378 IC50 = 7500 nM T15439 CPAU45 44383557 IC50 = 54000 nM T15439 CV13QW 44383558 IC50 = 8000 nM T15439 C6OXP9 44383561 IC50 = 9000 nM T15439 CA8MJ7 44383980 IC50 = 1000 nM T15439 C3XK4L 44384139 IC50 = 1000 nM T15439 CQ76HO 44384193 IC50 = 3000 nM T15439 CCD43W 44384304 IC50 = 30000 nM T15439 CDUN52 44384305 IC50 = 9000 nM T15439 C12REV 44384385 IC50 = 9000 nM T15439 CANV51 44384438 IC50 = 4500 nM T15439 CL7QI6 44416525 IC50 = 45 nM T15439 CKX67V 44416526 IC50 = 146 nM T15439 C8HC6X 44416527 IC50 = 300 nM T15439 C3OU9B 44416533 IC50 = 107 nM T15439 C8TJ0K 44416733 IC50 = 19 nM T15439 C3JK6V 44417104 IC50 = 535 nM T15439 CXW34I 44417113 IC50 = 190 nM T15439 C2HU1Z 44417114 IC50 = 463 nM T15439 CF2B7K 44417116 IC50 = 31 nM T15439 CEI6S5 44417117 IC50 = 63 nM T15439 C9DZ7B 44417118 IC50 = 27 nM T15439 CI37CH 44417122 IC50 = 116 nM T15439 CD0N8O 44417123 IC50 = 60 nM T15439 CFQ1X6 44417124 IC50 = 71 nM T15439 CDV29A 44417129 IC50 = 8700 nM T15439 CCFZ48 44417130 IC50 = 18 nM T15439 CR7BY2 44417153 IC50 = 50 nM T15439 CE3Q0O 44417158 IC50 = 54 nM T15439 C0JZ4C 44417159 IC50 = 57 nM T15439 CFED63 44417160 IC50 = 38 nM T15439 C0ID8W 44417199 IC50 = 23000 nM T15439 C1W7JC 44417200 IC50 = 25 nM T15439 CV58SG 44417205 IC50 = 100000 nM T15439 C8KD3J 44417206 IC50 = 6900 nM T15439 CD29CK 44417227 IC50 = 76 nM T15439 C58PXI 44448386 IC50 = 1900 nM T15439 CSI3H4 44448415 IC50 = 820 nM T15439 C8FM7R 44450395 IC50 > 10000 nM T15439 CAD15P 44450396 IC50 > 10000 nM T15439 CX54WI 44450403 IC50 > 10000 nM T15439 CKBH61 44450404 IC50 > 10000 nM T15439 C2XK3U 44450405 IC50 > 10000 nM T15439 C0G2DZ 44450406 IC50 > 10000 nM T15439 CT06GI 44450415 Ki = 8300 nM T15439 CR1FM5 44450416 IC50 > 10000 nM T15439 C3FX7L 44450417 IC50 > 10000 nM T15439 CY51GX 44450426 IC50 > 10000 nM T15439 CF17EP 44450439 IC50 > 10000 nM T15439 CLV38B 44450446 IC50 > 10000 nM T15439 CSX9T4 44450456 IC50 > 10000 nM T15439 CID60S 44450457 IC50 > 10000 nM T15439 CV2P8R 44450458 IC50 > 10000 nM T15439 CN6XM9 44450467 IC50 > 10000 nM T15439 CE06GZ 44450488 IC50 > 10000 nM T15439 CM0SP7 44567879 IC50 > 10000 nM T15439 CIJ0N7 44567913 IC50 > 10000 nM T15439 CV32CF 44567970 IC50 > 10000 nM T15439 CP4I5X 44567971 IC50 = 7400 nM T15439 CBN84U 44568046 IC50 > 10000 nM T15439 CR5L6E 44568047 IC50 > 10000 nM T15439 C4NP2D 44568090 IC50 = 380 nM T15439 CYFO65 44568091 IC50 > 10000 nM T15439 CNG7Z5 44568130 IC50 > 10000 nM T15439 CWDA52 44568131 IC50 > 10000 nM T15439 C86IZV 44568165 IC50 > 10000 nM T15439 CVY97F 44568166 IC50 > 10000 nM T15439 CXV3I6 44581449 IC50 = 3 nM T15439 CKI6S0 44581481 IC50 > 1000 nM T15439 C73AWH 44581482 IC50 = 15 nM T15439 C37UCL 44581483 IC50 = 350 nM T15439 C2L0EX 44581484 IC50 = 8 nM T15439 C2JS7Q 44581545 IC50 = 12 nM T15439 CT8Z4K 44581546 IC50 = 45 nM T15439 CAF9Z3 44581547 IC50 = 25 nM T15439 CZ4I3G 44581572 IC50 > 1000 nM T15439 CMP1H4 44581573 IC50 = 200 nM T15439 COT17R 44581574 IC50 = 500 nM T15439 C9FVK0 44581575 IC50 = 90 nM T15439 CA3Y0D 44581615 IC50 = 500 nM T15439 C8D0GS 44581616 IC50 = 47 nM T15439 CD7FM9 44581617 IC50 > 1000 nM T15439 CLSO84 44581650 IC50 > 1000 nM T15439 CG4FT8 44581651 IC50 > 1000 nM T15439 CT5F9X 44581652 IC50 = 790 nM T15439 C8VT9H 44581653 IC50 = 325 nM T15439 CXS0Z7 44589629 IC50 = 1000 nM T15439 CC7Z5W 44589630 IC50 = 330 nM T15439 C01SWN 44589666 IC50 = 200 nM T15439 CBY26Z 44589667 IC50 > 1000 nM T15439 C6QWD4 44589668 IC50 = 350 nM T15439 CAP4K2 44589669 IC50 = 70 nM T15439 CN9L6Q 44589704 IC50 = 75 nM T15439 C8X5PR 44589705 IC50 > 1000 nM T15439 CI4NQ2 44589706 IC50 > 1000 nM T15439 CG9WX7 44589707 IC50 = 175 nM T15439 CSX1G9 44589742 IC50 = 370 nM T15439 CO93SH 44589743 IC50 = 5 nM T15439 C69RYZ 44589744 IC50 > 1000 nM T15439 CDI78W 44589781 IC50 > 1000 nM T15439 C2OAD8 44589782 IC50 = 1000 nM T15439 C28QPO 44589783 IC50 = 80 nM T15439 CE0JI6 44589784 IC50 > 1000 nM T15439 CNVA28 44589817 IC50 = 835 nM T15439 CDHK69 44589818 IC50 = 175 nM T15439 CG9V3Y 44589819 IC50 = 1.5 nM T15439 C86FTU 44589820 IC50 = 18 nM T15439 CQ54PU 44589862 IC50 = 400 nM T15439 CSOE13 44589863 IC50 = 110 nM T15439 C96FOQ 44589864 IC50 = 300 nM T15439 CASQ04 44589865 IC50 = 35 nM T15439 C9D6YM 44589919 IC50 > 1000 nM T15439 CHB0V5 44589920 IC50 = 395 nM T15439 C2SB3O 44589921 IC50 = 90 nM T15439 CY8L7K 44589922 IC50 = 435 nM T15439 CPW64I 44589976 IC50 = 5 nM T15439 C7PUR0 44589977 IC50 = 89 nM T15439 C0N1KC 44589978 IC50 = 290 nM T15439 C7ER1D 44590340 IC50 = 1000 nM T15439 CR9MF1 44590341 EC50 = 123.03 nM T15439 CTV9J3 44590401 IC50 > 10000 nM T15439 CP30EL 44590402 IC50 > 10000 nM T15439 CS58YP 44590403 IC50 = 794.33 nM T15439 CA49GO 44590404 IC50 > 10000 nM T15439 C3RH8X 44590445 IC50 = 63.1 nM T15439 CP9SU5 44590446 IC50 > 100 nM T15439 CXOC39 44590447 IC50 = 19.95 nM T15439 CVL1S9 44590448 IC50 = 39.81 nM T15439 CWVR62 44590515 IC50 = 100 nM T15439 CJ17UF 44590516 IC50 = 199.53 nM T15439 CZ93YT 44590517 IC50 = 316.23 nM T15439 CA6BM0 44590518 IC50 = 3162.28 nM T15439 C4GR0W 44593654 IC50 = 31 nM T15439 C0PQA1 46225376 EC50 > 60000 nM T15439 C2O1HF 46225392 EC50 > 60000 nM T15439 C2KJV1 46225393 IC50 > 60000 nM T15439 CK8QW4 46225413 IC50 = 400 nM T15439 CW78DI 49799080 IC50 = 501.19 nM T15439 C8PH3O 49799081 IC50 = 1995.26 nM T15439 CO48HR 49799082 IC50 = 29000 nM T15439 C2ANS9 73345497 Ki = 200 nM T15439 CX2Z7N 73354472 Ki = 150000 nM T15439 CX3SC2 100972207 IC50 = 4786.3 nM T15439 CM20FH 100972208 IC50 = 794.33 nM T15439 CM31ZT 118719096 Ki = 600000 nM T15439 C60AYU 118719108 IC50 = 3000 nM T15439 CA2P9V 118719109 IC50 > 173.78 nM T15439 C2N9JO 118719110 IC50 = 1200 nM T15439 D00HAJ 73347136 IC50 = 39 nM T15439 D03QAN 71166 IC50 = 3.3 ug.mL-1 T15439 D03TBA 10020451 IC50 = 800 nM T15439 D04JXA 5311122 IC50 = 3 nM T15439 D09MAZ 46897162 IC50 > 5000 nM T15439 D0J3FH 10218379 Ki = 15.2 nM T15851 C3R2CQ 150856 Ki = 98000 nM T15851 CGS97U 71513567 Ki = 28300 nM T15851 CRZU86 135566518 Ki = 17 nM T15851 CRAO63 145948304 Ki > 4000000 nM T15851 C4HID1 145948305 Ki = 759000 nM T15851 CM8P3U 145948306 Ki > 2000000 nM T15851 D00GOC 135413551 Ki = 17 nM T15851 D08OFS 16666489 Ki = 18200 nM T15851 D0C7PT 16666487 Ki = 16600 nM T15851 D0DW2F 16124514 Ki = 1100 nM T15851 D0H9DJ 6030 Ki = 220000 nM T15851 D0P7AS 25027092 Ki = 350 nM T15851 D0S2QZ 6131 Ki = 1400000 nM T43548 CA7H1P 788151 IC50 = 120000 nM T43548 C2YUR1 3800971 IC50 = 212000 nM T43548 C7EL1A 22433034 IC50 = 70000 nM T43548 C8AK6R 72105690 IC50 = 86000 nM T43548 C7L6TF 80763614 IC50 = 4960 nM T43548 C6V0AD 135385826 IC50 = 150 nM T43548 CJ4E6T 135385997 IC50 = 1400 nM T43548 CO4V8E 135386034 IC50 = 710 nM T43548 CAO8P9 135386050 IC50 = 86 nM T43548 CH5D1Q 135386055 IC50 = 710 nM T43548 CG5HM7 135386075 IC50 = 390 nM T43548 CTIF48 135386175 IC50 = 230 nM T43548 C81YSO 135386184 IC50 = 640 nM T43548 CVGR85 135386269 IC50 = 3500 nM T43548 CZ43RM 135386310 IC50 = 2500 nM T43548 CFN6A5 135386315 IC50 = 680 nM T43548 CPTO52 135386361 IC50 = 400 nM T43548 C1Z9NH 135386376 IC50 = 2100 nM T43548 CAQ0P3 135386382 IC50 = 990 nM T43548 CR2B7X 135386383 IC50 = 260 nM T43548 CDQX16 135386741 IC50 = 1700 nM T43548 CEHY16 135386838 IC50 = 430 nM T43548 C8AV1D 135386844 IC50 = 1000 nM T43548 C6CLQ5 135386845 IC50 = 330 nM T43548 CL9UH2 135386854 IC50 = 1200 nM T43548 CP79GZ 135386866 IC50 = 860 nM T43548 C17NVH 135386892 IC50 = 960 nM T43548 CX95CB 135386897 IC50 = 930 nM T43548 CU59MD 135386899 IC50 = 200 nM T43548 CX6DT2 135386909 IC50 = 790 nM T43548 CA0MD2 135386920 IC50 = 130 nM T43548 CK3FI8 135386935 IC50 = 1900 nM T43548 C0RH2L 135386938 IC50 = 520 nM T43548 CUOE02 135386944 IC50 = 3900 nM T43548 C4KMN5 135386972 IC50 = 97 nM T43548 CU9PD5 135387021 IC50 = 3400 nM T43548 C7SO4L 135387022 IC50 = 400 nM T43548 CB8H7T 135387414 IC50 = 37000 nM T43548 C5TYP2 135747590 IC50 = 27000 nM T43548 CJ1IS2 135886621 IC50 > 31622.78 nM T43548 CV96BZ 137348674 IC50 = 480 nM T43548 C4K3HX 137348712 IC50 = 2.9 nM T43548 C9ZQW1 137348715 IC50 = 350 nM T43548 CD2FR4 137551963 IC50 = 142000 nM T43548 C6IWZ7 137631722 IC50 = 1.7 nM T43548 C0FUL9 137631964 IC50 = 2300 nM T43548 CO8CY1 137634100 IC50 = 61000 nM T43548 CZW72J 137634597 IC50 > 99000 nM T43548 C2G5IW 137634601 IC50 = 6100 nM T43548 C8RYA2 137634921 IC50 = 11 nM T43548 CQSE49 137636045 IC50 > 100000 nM T43548 C23TJX 137637495 IC50 = 590 nM T43548 C3NEB1 137637555 IC50 = 398.11 nM T43548 CC4F6Y 137639165 IC50 = 390 nM T43548 COR6U1 137640061 IC50 = 210 nM T43548 CJF6A2 137640382 IC50 = 212000 nM T43548 CIL20W 137641266 IC50 = 125.89 nM T43548 C7CB2D 137643992 IC50 = 64000 nM T43548 C7SA9V 137644739 IC50 = 1.5 nM T43548 C8H2LK 137644920 IC50 = 24000 nM T43548 CDV7C5 137645207 IC50 = 0.87 nM T43548 C1B5RH 137646123 IC50 = 45000 nM T43548 COS8I0 137646360 IC50 > 10000 nM T43548 C4U7QT 137646364 IC50 = 24 nM T43548 CUFW31 137646739 IC50 = 55 nM T43548 CTUQ83 137647013 IC50 = 29 nM T43548 CCE1Z0 137649341 IC50 = 370 nM T43548 C8WUN1 137650966 IC50 = 1 nM T43548 CA9P2Y 137651007 IC50 = 36 nM T43548 C5R1FA 137652065 IC50 = 8200 nM T43548 CV9U3G 137653457 IC50 > 99000 nM T43548 C25MDP 137654713 IC50 = 2.4 nM T43548 CDE49N 137655163 IC50 = 15 nM T43548 C1MU7K 137656202 IC50 = 5 nM T43548 C3WQL8 137656281 IC50 = 12 nM T43548 CP4UZ3 137657955 IC50 = 16 nM T43548 CA6GZ1 137659373 IC50 = 3.3 nM T43548 C30KIH 137660565 IC50 = 2900 nM T43548 C1M7HV 137661449 IC50 = 13 nM T43548 C64UPR 142478626 IC50 = 190 nM T43548 C7E9AW 142478649 IC50 = 480 nM T43548 C3JFU7 142478704 IC50 = 1400 nM T43548 CO53XV 145950480 IC50 = 62000 nM T43548 C7L3NA 145953045 IC50 = 112000 nM T43548 CMP41A 145955890 IC50 = 34000 nM T43548 CQHS73 145959063 IC50 = 80000 nM T43548 CC23GU 145971457 IC50 = 170000 nM T43548 CAQD05 146020593 IC50 = 207000 nM T43548 CM21QX 146020594 IC50 = 3400 nM T43548 C52CYT 146020597 IC50 = 4500 nM T43548 CAGL36 146035908 IC50 = 4600 nM T43548 CIML61 151934891 IC50 = 760 nM T43548 C70RTH 151960901 IC50 = 270 nM T43548 CN01XI 152233765 IC50 = 310 nM T43548 C0VNT5 155517294 IC50 = 890 nM T43548 C0SQ4X 155518342 IC50 = 2440 nM T43548 CR21IZ 155518808 IC50 = 770 nM T43548 CVK7G4 155519879 IC50 = 25 nM T43548 CM0OE9 155520643 IC50 = 9560 nM T43548 C2VM0G 155524175 IC50 = 3440 nM T43548 C8BW5I 155524510 IC50 = 1120 nM T43548 CZ4CG7 155525789 IC50 = 1040 nM T43548 CJK2X7 155525999 IC50 = 520 nM T43548 C0V9RE 155526027 IC50 > 20000 nM T43548 CCO35B 155526202 IC50 = 2040 nM T43548 C6DOM9 155528623 IC50 = 4220 nM T43548 C6LEO3 155529082 IC50 = 14900 nM T43548 CBQH32 155533638 IC50 = 1850 nM T43548 CL4AI2 155536551 IC50 = 6600 nM T43548 CW7CR8 155537417 IC50 = 2460 nM T43548 CN1K7A 155538022 IC50 = 7410 nM T43548 CM0UF7 155538999 IC50 = 1850 nM T43548 C8WAN1 155540902 IC50 = 190 nM T43548 C5K8XV 155541010 IC50 = 4830 nM T43548 C18PQF 155543278 IC50 = 5400 nM T43548 C1OZ9W 155545492 IC50 = 980 nM T43548 C4G7DF 155546160 IC50 = 860 nM T43548 C4K1LI 155549001 IC50 = 470 nM T43548 CBSM80 155549668 IC50 = 7720 nM T43548 CQVL35 155550865 IC50 > 10000 nM T43548 C23NCJ 155550965 IC50 = 1730 nM T43548 CU3ZP0 155551469 IC50 > 10000 nM T43548 C6XCZ2 155552228 IC50 > 20000 nM T43548 CLN1A6 155552783 IC50 = 17300 nM T43548 C6M1FP 155558661 IC50 > 10000 nM T43548 C7C6RO 155559510 IC50 > 10000 nM T43548 CSOE83 155559582 IC50 = 4850 nM T43548 CH4RZ1 155561643 IC50 > 10000 nM T43548 CSQE74 155568277 IC50 = 2590 nM T02777 D02KMO 4826 EC50 = 3540 nM T02777 D00LWF 43345 EC50 = 230 nM T02777 CRN4U9 443423 EC50 = 1250 nM T02777 C3EMG9 15953834 EC50 = 750 nM T02777 CW8AL1 20246092 EC50 = 21100 nM T02777 C74QXU 42609940 EC50 = 670 nM T02777 CET0X3 44564052 EC50 = 2600 nM T02777 CRT8S9 44564053 EC50 = 8440 nM T02777 CBRG65 44564087 EC50 = 3090 nM T02777 CGV0C4 44564088 EC50 = 16500 nM T02777 CLQ7S6 44564089 EC50 = 310 nM T02777 C23SBW 44564125 EC50 = 120 nM T02777 C46WHS 44564126 EC50 = 2070 nM T02777 CSV8N2 44564127 EC50 = 70 nM T02777 C74FAM 44564128 EC50 = 780 nM T02777 C14VFK 44564182 EC50 = 810 nM T02777 CX19UC 44564183 EC50 = 7060 nM T02777 CV0K2S 44564184 EC50 = 560 nM T02777 C6LZG1 44564185 EC50 = 1540 nM T02777 CASW43 44564186 EC50 = 18600 nM T02777 CX15FG 44564202 EC50 = 1500 nM T02777 CK1MC6 44564203 EC50 = 2750 nM T02777 C6G9QC 44564204 EC50 = 7450 nM T02777 CE08SN 44564205 EC50 > 30000 nM T02777 CN36YV 44564206 EC50 = 13000 nM T02777 C9C4SV 44564249 EC50 > 30000 nM T02777 CN81XK 44564250 EC50 = 12900 nM T02777 CPB08Q 44564251 EC50 = 4330 nM T02777 C62AXW 44564252 EC50 = 1640 nM T02777 C2DLQ6 44564253 EC50 = 13800 nM T02777 C2XFE1 44564292 EC50 = 14700 nM T02777 CCV9S5 44564293 EC50 = 7850 nM T02777 CI50RA 44564294 EC50 = 16100 nM T02777 CJ3C2A 44564295 EC50 = 6180 nM T02777 C3I0QC 44564321 EC50 = 6850 nM T02777 C8Q7UY 44564322 EC50 = 1370 nM T02777 CZ4LK1 44564323 EC50 = 7770 nM T02777 CZ2TS5 44564324 EC50 > 30000 nM T02777 CLK06R 44564347 EC50 = 24800 nM T02777 CZ9G6J 44564348 EC50 = 20400 nM T02777 CX71IQ 44564349 EC50 = 6940 nM T02777 CGB80T 44564350 EC50 = 2440 nM T02777 C5KTZ9 44564386 EC50 = 14100 nM T02777 CAN49I 44564387 EC50 = 4100 nM T02777 CR6EZ8 44564388 EC50 = 1560 nM T02777 COY63I 44564422 EC50 = 1080 nM T02777 C5VL8Q 44564423 EC50 = 820 nM T02777 CX67CV 44564424 EC50 = 10300 nM T02777 CMHZ03 44564425 EC50 = 6450 nM T02777 C7KG4E 44564464 EC50 = 7330 nM T02777 C48WVY 44564465 EC50 = 7990 nM T02777 CVTR92 44564466 EC50 = 1710 nM T02777 CW25EZ 44564467 EC50 = 3160 nM T02777 CEN31X 44564513 EC50 = 6040 nM T02777 CDF34K 136036211 EC50 = 2290 nM T02777 C65IVR 136036217 EC50 = 3710 nM T81443 D0W9LX 2585 IC50 = 32220 nM T81443 D0E4GG 11703255 IC50 = 680 nM T81443 D0SJ8Q 6912404 IC50 = 1.5 nM T81443 CB9I6Y 2534913 IC50 = 167500 nM T81443 CJ8PL6 4840815 IC50 = 34170 nM T81443 CGO2I1 8087741 IC50 = 64100 nM T81443 CP3QT1 9560223 IC50 = 164000 nM T81443 CG80YR 9863761 IC50 = 160 nM T81443 CT7JC1 9919285 IC50 = 3.2 nM T81443 CG4M6C 11516340 IC50 = 240 nM T81443 C6AF1V 11552188 IC50 > 10000 nM T81443 CO6Q7D 11562896 IC50 = 4500 nM T81443 CUG85Z 11645958 IC50 = 110 nM T81443 C2HMR0 16247145 IC50 = 16600 nM T81443 CA0GC9 44405661 IC50 = 250 nM T81443 C12EAM 44405768 IC50 = 160 nM T81443 C0Q5XC 44405780 IC50 = 80 nM T81443 CBZ97N 44405822 IC50 = 350 nM T81443 C63JNA 44408420 IC50 = 175000 nM T81443 CC96NU 44408426 IC50 = 35600 nM T81443 CG9A3Z 44408517 IC50 = 61400 nM T81443 C8GFB1 44408519 IC50 = 27600 nM T81443 C1OAW5 44408521 IC50 = 9400 nM T81443 CPW68S 44408523 IC50 = 10500 nM T81443 CA56LB 44408634 IC50 = 6110 nM T81443 C9F4DR 44408639 IC50 = 190000 nM T81443 C3OQ8N 44589052 IC50 > 10000 nM T81443 CEXM35 44589758 IC50 = 5.3 nM T81443 C5TR7E 66573231 EC50 = 3950 nM T81443 CE57XK 71158523 IC50 = 32550 nM T81443 CH29GF 71258526 IC50 > 10000 nM T81443 CUNZ36 71682591 EC50 = 8260 nM T81443 CDV5S0 71718403 IC50 = 1.5 nM T81443 CA0CF5 73774537 IC50 = 7700 nM T81443 C4I0OG 78426192 EC50 = 3900 nM T81443 C3IO1J 78426193 EC50 = 390 nM T81443 CL4W5I 90655905 EC50 = 790 nM T81443 CF63UP 90655906 EC50 = 2000 nM T81443 C3BYV9 90655907 EC50 = 2000 nM T81443 CLKN01 90655908 EC50 > 10000 nM T81443 CZ72PU 90655909 EC50 = 1000 nM T81443 CP68NB 90655910 EC50 = 6300 nM T81443 CU2B3R 90655911 EC50 = 3900 nM T81443 CQH90B 90655912 EC50 = 500 nM T81443 C90UND 90655913 EC50 = 790 nM T81443 C7CK4M 90655914 EC50 = 630 nM T81443 CWB57V 90655915 EC50 = 630 nM T81443 CUG7Z5 90655916 EC50 = 3900 nM T81443 C9RJ8T 90655917 EC50 = 630 nM T81443 C1JXR2 90655918 EC50 = 2000 nM T81443 CI6AJ1 90655919 EC50 = 1200 nM T81443 CFQ30V 90655920 EC50 = 10000 nM T81443 CT28LE 90655921 EC50 = 7900 nM T81443 CX4HU5 90655922 EC50 = 5000 nM T81443 C5MZW6 90655923 EC50 = 2500 nM T81443 CH90DR 90655924 EC50 = 2000 nM T81443 CW17KR 90655925 EC50 = 3100 nM T81443 CQO87B 90655926 EC50 = 3100 nM T81443 C7C9KU 90655927 EC50 = 3100 nM T81443 CKDY39 90655928 EC50 = 7900 nM T81443 C3H9EW 90655929 EC50 = 3100 nM T81443 CC7W9M 90655930 EC50 = 3100 nM T81443 C1BV8R 90655931 EC50 = 790 nM T81443 CIW60O 90655932 EC50 = 1000 nM T81443 CW60LJ 90655933 EC50 = 2500 nM T81443 CQ5J9M 90655934 EC50 > 10000 nM T81443 CZI15M 90655935 EC50 > 10000 nM T81443 C4X9TN 90655936 EC50 > 10000 nM T81443 C2V3KB 90655937 EC50 > 10000 nM T81443 CY9N1V 90655938 EC50 = 3100 nM T81443 C9PGU8 90655939 EC50 = 15800 nM T81443 C47XFO 90655940 EC50 = 3100 nM T81443 CHJ0Z9 90655941 EC50 = 3100 nM T81443 CU3GI8 90655942 EC50 = 3900 nM T81443 CKE53L 90655943 EC50 = 3100 nM T81443 CLS4I1 90655944 EC50 > 10000 nM T81443 C6KOD5 90655945 EC50 > 10000 nM T81443 C4X0JN 90655946 EC50 > 10000 nM T81443 C78SOE 90655947 EC50 = 1200 nM T81443 C7E3FJ 90655948 EC50 = 790 nM T81443 CS3Y9T 90655949 EC50 = 3100 nM T81443 CG86XI 101882318 EC50 = 0.4 nM T81443 CESN49 101882319 EC50 = 0.08 nM T81443 C58ERK 101882320 EC50 = 31 nM T81443 CU8C0A 118724518 IC50 = 3700 nM T81443 CU6GV9 118724526 IC50 = 1300 nM T81443 CB7VO2 118724528 IC50 = 5000 nM T81443 CK03YN 118724530 IC50 = 200 nM T81443 CW6UQ0 132502975 EC50 = 3270 nM T81443 C45BQH 132585194 EC50 > 100000 nM T81443 CWV63A 134129840 IC50 = 1230 nM T81443 C12WYF 136179591 IC50 = 59100 nM T81443 CA5JQ3 137632780 EC50 = 3270 nM T81443 CH40RS 137633058 EC50 = 430 nM T81443 CI64KV 137634073 EC50 > 10000 nM T81443 CO5AQ1 137635519 EC50 = 11080 nM T81443 C0QOL5 137636236 EC50 > 10000 nM T81443 CMB21V 137636834 EC50 > 10000 nM T81443 CXCL56 137636966 EC50 > 10000 nM T81443 CY2ZC8 137637513 EC50 > 10000 nM T81443 C0IK7F 137638193 IC50 = 630 nM T81443 C1NBH3 137638254 EC50 = 4900 nM T81443 CU2FH9 137638726 EC50 = 3750 nM T81443 CZ6H0V 137639041 IC50 = 5450 nM T81443 CRH6O5 137641475 EC50 = 6350 nM T81443 CBF45N 137641507 EC50 > 10000 nM T81443 CW5CH7 137641887 EC50 > 10000 nM T81443 CRP1V8 137642610 EC50 > 10000 nM T81443 C62LIR 137643594 EC50 > 10000 nM T81443 CCTU29 137644858 EC50 > 10000 nM T81443 CZV34Q 137646359 EC50 = 14000 nM T81443 CYVC34 137647919 EC50 = 11680 nM T81443 CV3S6W 137647950 EC50 > 10000 nM T81443 CCO6F0 137648018 EC50 > 10000 nM T81443 CDW7L6 137649081 EC50 > 10000 nM T81443 C2VYA6 137651264 EC50 = 2120 nM T81443 C6CN0B 137651794 EC50 = 7420 nM T81443 CY3O6Z 137651902 EC50 > 10000 nM T81443 CQ3TU5 137652008 EC50 > 10000 nM T81443 CHA97O 137652867 EC50 > 10000 nM T81443 CK1S3N 137652884 EC50 > 10000 nM T81443 CPRW87 137655143 EC50 > 10000 nM T81443 CA6O0B 137656090 EC50 > 10000 nM T81443 CY59VS 137657271 EC50 > 10000 nM T81443 CX72LT 137657449 EC50 = 920 nM T81443 CERM92 137658225 EC50 > 10000 nM T81443 CM0HF9 137658681 EC50 = 3580 nM T81443 CFS6R4 137659575 EC50 = 12000 nM T81443 C7Y3VO 137660059 EC50 > 10000 nM T81443 CGJ87K 137661578 EC50 > 10000 nM T81443 CA1O9E 141761144 IC50 = 31540 nM T81443 C9N4OB 141761145 IC50 = 13640 nM T81443 C98EHJ 141761146 IC50 = 34640 nM T81443 CA4NT8 141761147 IC50 = 15110 nM T81443 CF7SW6 141761150 IC50 = 12450 nM T81443 C97KQW 141761151 IC50 = 24680 nM T81443 C6FEI9 141761152 IC50 = 16680 nM T81443 CJ20AX 141761153 IC50 = 55390 nM T81443 CR7AU2 141761155 IC50 = 51540 nM T81443 C9J0DW 141761156 IC50 = 54600 nM T81443 CT4VS9 145950641 IC50 = 26020 nM T81443 CKC26Y 145951568 IC50 = 21120 nM T81443 C37SZW 145954440 IC50 = 12390 nM T81443 C08WEU 145955041 IC50 = 28530 nM T81443 CN4JV9 145958212 IC50 = 21710 nM T81443 C2EMT8 145960309 IC50 = 25920 nM T81443 CTP64Q 145967497 IC50 = 540 nM T81443 CB53JT 145967694 IC50 = 19250 nM T81443 CR1LX0 145969011 IC50 = 45650 nM T81443 CKBI34 145988409 IC50 = 5420 nM T81443 CRX3V8 145989045 IC50 = 25900 nM T81443 CFK28P 155511732 IC50 = 5000 nM T81443 C4SOZ0 155512070 IC50 = 3897 nM T81443 CE5P4K 155521327 IC50 = 334 nM T81443 CZ9TN6 155529716 IC50 = 20000 nM T81443 CV3L5G 155549519 IC50 = 1785 nM T81443 C96GUM 155560601 IC50 = 2701 nM T81443 D06MKE 24849153 IC50 = 2.4 nM T81443 D0J0GM 44224215 IC50 = 3000 nM T39380 CD2K9I 219925 IC50 > 9400 nM T39380 CNX1I9 744590 Ki = 20.8 nM T39380 C4ESQ9 1105689 Ki = 21.1 nM T39380 C4TGR0 2260227 Ki = 7.2 nM T39380 C32MJD 3114900 EC50 = 3300 nM T39380 CN8XM2 5311263 EC50 = 2 nM T39380 CAX9U1 5473680 EC50 > 11400 nM T39380 CDM1E9 5861754 IC50 = 355 nM T39380 CLS96Y 6419701 EC50 = 288.4 nM T39380 C1K9GW 9824415 IC50 = 260 nM T39380 CA78VE 9958483 IC50 > 50000 nM T39380 C7B8UT 10126584 IC50 = 55 nM T39380 CG65LQ 10126736 IC50 = 420 nM T39380 CCG97S 10127776 IC50 = 80 nM T39380 C8IGL1 10136738 EC50 = 1089 nM T39380 CGCK28 10149985 IC50 = 26 nM T39380 C3LG4R 10150372 IC50 = 32 nM T39380 CPU38H 10151146 IC50 = 6.6 nM T39380 CDE1S4 10172354 IC50 = 530 nM T39380 CI5X6K 10172513 IC50 = 250 nM T39380 CWJO04 10172546 IC50 = 74 nM T39380 CS62VA 10173002 IC50 = 89 nM T39380 CL2QV0 10173327 IC50 = 57 nM T39380 C8XZV1 10174548 IC50 = 42 nM T39380 CR9YM8 10193915 IC50 = 59 nM T39380 C56XBS 10215741 IC50 = 700 nM T39380 CKPV49 10287091 IC50 = 2100 nM T39380 C74CKG 10287343 IC50 = 450 nM T39380 CW5JG7 10287365 IC50 = 120 nM T39380 C3R1AI 10288370 IC50 = 33 nM T39380 C6EY2U 10289318 IC50 = 23 nM T39380 C8VP3G 10309271 IC50 = 1200 nM T39380 C7B2FU 10309462 IC50 = 15 nM T39380 CAF85E 10310253 IC50 = 36 nM T39380 C8HBY4 10311227 IC50 = 18 nM T39380 COZF72 10322404 EC50 = 112 nM T39380 CIF3K9 11312936 EC50 = 2500 nM T39380 CQLP42 11473989 EC50 = 244 nM T39380 CFHV74 11568387 EC50 = 6330 nM T39380 C0CBY2 11625765 EC50 = 5720 nM T39380 C7QRT8 11648176 EC50 = 100 nM T39380 CY3L7V 11755685 EC50 ~ 11000 nM T39380 CZO6H5 16045222 EC50 = 7170 nM T39380 C05BUC 23701125 EC50 = 1710 nM T39380 CJ5OV6 23701126 EC50 = 1170 nM T39380 C1F9GI 24882686 IC50 = 17 nM T39380 C4F8UE 44343851 EC50 > 5000 nM T39380 CD1SX3 44343866 EC50 = 108 nM T39380 CK0NG4 44343867 EC50 > 5000 nM T39380 C5J4BE 44343880 EC50 = 1960 nM T39380 CS7BJ1 44344023 EC50 > 5000 nM T39380 C31BXA 44344270 IC50 = 120 nM T39380 CY7FC4 44344298 IC50 = 270 nM T39380 CV86RF 44368508 EC50 = 147.91 nM T39380 CPS46Q 44406620 EC50 = 1320 nM T39380 CL3FU4 44406630 Ki = 745 nM T39380 CIX30G 44406632 EC50 > 10000 nM T39380 CS28VK 44406644 EC50 = 1300 nM T39380 CYUF09 44406648 EC50 = 1170 nM T39380 CO1GB3 44406649 EC50 = 1710 nM T39380 C3ZTC9 44406674 EC50 = 1090 nM T39380 C7DY4Q 44406675 EC50 > 10000 nM T39380 C91BKR 44406679 EC50 = 1540 nM T39380 C3SX2V 44414935 EC50 > 9460 nM T39380 C2WEQ7 44437392 IC50 = 40000 nM T39380 CP1FN6 44437417 IC50 = 6000 nM T39380 C29TWV 44454059 IC50 = 260 nM T39380 CLU5R6 44454091 IC50 = 35 nM T39380 CV13MG 44454136 IC50 = 170 nM T39380 CB19QS 44454163 IC50 = 310 nM T39380 CNVI84 44454164 IC50 = 1860 nM T39380 C3VI5O 44454165 IC50 = 730 nM T39380 C7KY2V 44454191 IC50 = 6610 nM T39380 C3Z1BK 44454215 IC50 = 730 nM T39380 CL7DB5 44454216 IC50 > 30000 nM T39380 CVP0H5 44454245 IC50 > 30000 nM T39380 C0XH1N 44454246 IC50 > 30000 nM T39380 CI15RQ 44454274 IC50 > 30000 nM T39380 C93RQI 44454305 IC50 = 1300 nM T39380 CA5Y1E 44454306 IC50 = 3200 nM T39380 CO7L3S 44454369 IC50 > 50000 nM T39380 C5L0ZB 44454370 IC50 = 1700 nM T39380 C85ANH 46213949 IC50 > 8000 nM T39380 CET63X 46223906 EC50 = 161 nM T39380 C8CK4M 46240292 IC50 = 1700 nM T39380 CWF21Q 66552906 IC50 > 10000 nM T39380 C9GQ2D 66774612 IC50 = 23000 nM T39380 CW2O5R 66774777 IC50 = 790 nM T39380 CKL76D 66775043 IC50 = 8600 nM T39380 C57TYK 71569053 EC50 = 114.82 nM T39380 CSN3I7 71569056 EC50 = 146 nM T39380 CPT5S2 71718248 EC50 = 117 nM T39380 CKC4U7 71719457 EC50 = 350 nM T39380 C5P1CQ 71720690 EC50 = 109.65 nM T39380 CC2BA0 73053706 EC50 = 2160 nM T39380 CW7BX6 73296090 EC50 = 50 nM T39380 C4C7TR 73296091 EC50 = 3600 nM T39380 CKH6F0 73296092 EC50 = 110 nM T39380 C7KB2X 73296094 EC50 = 1420 nM T39380 CR32EN 77461257 EC50 = 0.00506 nM T39380 CL3Y8J 89484779 IC50 > 800 nM T39380 CQ3PK4 90308914 IC50 > 800 nM T39380 C89FXZ 90309040 IC50 > 800 nM T39380 CYSQ05 90309100 IC50 > 800 nM T39380 CY3ZT1 90309524 IC50 > 800 nM T39380 C42IJD 118710194 EC50 = 60 nM T39380 CFLV86 118710197 EC50 = 0.15 nM T39380 CNI96W 118728428 IC50 > 25000 nM T39380 C3O6KB 118728429 IC50 > 26000 nM T39380 C4U3DG 118728430 IC50 > 800 nM T39380 C8U0GE 118728431 IC50 > 800 nM T39380 C72NCP 118728432 IC50 > 25000 nM T39380 C2YHT8 118728433 IC50 > 25000 nM T39380 C4M3YA 118728434 IC50 > 25000 nM T39380 CG65XZ 122191108 Ki = 170 nM T39380 CKL42I 122191542 EC50 = 108 nM T39380 CWQ8Y3 122191544 IC50 = 1420 nM T39380 D02RYR 11447695 EC50 = 3800 nM T39380 D03HLU 11276402 EC50 > 10000 nM T39380 D04BLL 11312382 EC50 = 4100 nM T39380 D04KQT 10468943 EC50 = 1000 nM T39380 D05TVG 23682233 Ki = 170 nM T39380 D07WLV 11219269 EC50 = 717 nM T39380 D07YUV 11197104 EC50 = 397 nM T39380 D0BP3E 11393306 EC50 ~ 10000 nM T39380 D0D5QS 11725751 IC50 = 40 nM T39380 D0E0DY 62532 EC50 = 1800 nM T39380 D0F2SQ 11288209 EC50 > 10000 nM T39380 D0N4AG 11220562 EC50 = 480 nM T39380 D0P7GR 78401 Ki = 3550 nM T39380 D0R8LB 44343825 EC50 = 30 nM T39380 D0X0UR 5497152 EC50 = 3 nM T39380 D0XJ9P 75816 EC50 = 3100 nM T39380 D0XY0Z 11208266 EC50 = 677 nM T39380 D0Z2QV 11242245 EC50 = 4570 nM T85943 D01PZD 5329098 IC50 = 16400 nM T85943 D03MNN 11341869 IC50 = 15 nM T85943 D03ZBT 11626560 IC50 > 10000 nM T85943 D04LVK 57379345 IC50 = 1694 nM T85943 D06ACW 6083 IC50 = 100 nM T85943 D06XXH 11511120 IC50 = 110 nM T85943 D09KTS 24821094 IC50 = 38 nM T85943 D09XZB 123631 IC50 = 1100 nM T85943 D0AZ3C 5291 IC50 > 25000 nM T85943 D0B0AX 5328127 IC50 > 50000 nM T85943 D0C4RB 36314 IC50 > 10000 nM T85943 D0E6XR 3062316 Ki = 0.295 nM T85943 D0G6QF 3081361 IC50 = 44 nM T85943 D0H0EQ 24826799 IC50 = 2.5 nM T85943 D0IQ6P 25102847 IC50 = 178 nM T85943 D0J1MI 4030 IC50 > 10000 nM T85943 D0J9ZR 4477 IC50 = 10000 nM T85943 D0K8KX 5280343 IC50 = 120 nM T85943 D0N3UL 3418 IC50 = 2000000 nM T85943 D0OB0F 5328940 IC50 = 1 nM T85943 D0R0MW 5329102 IC50 = 152.8 nM T85943 D0W5HK 216239 IC50 = 390 nM T85943 D02LJW 23635314 IC50 = 6.5 nM T85943 D02NNV 3038525 IC50 > 5000 nM T85943 D02RID 11545920 IC50 = 67000 nM T85943 D02UFQ 11620908 IC50 > 10000 nM T85943 D03AND 11656518 IC50 > 10000 nM T85943 D03LWG 53235510 IC50 = 2969 nM T85943 D04AHQ 71721540 IC50 = 310 nM T85943 D05NFR 135565923 IC50 = 5.3 nM T85943 D05PZB 135398495 IC50 = 10 nM T85943 D07EHV 44814409 IC50 > 10000 nM T85943 D07HPJ 11476171 IC50 = 4000 nM T85943 D08AOZ 86582336 IC50 = 1100 nM T85943 D0CY1B 6420138 Ki = 820 nM T85943 D0E3TC 44259 IC50 = 0.83 nM T85943 D0FD6D 11751922 IC50 = 37 nM T85943 D0GP9Q 11973736 IC50 >= 10000 nM T85943 D0I6VU 176167 IC50 > 100000 nM T85943 D0L4FS 5280961 IC50 > 10000 nM T85943 D0LF1U 5287969 IC50 = 34000 nM T85943 D0M0XB 10302451 IC50 = 2.7 nM T85943 D0M9QZ 11485656 IC50 = 50000 nM T85943 D0O6WV 24794418 IC50 > 500 nM T85943 D0P6DJ 151194 IC50 > 10000 nM T85943 D0Q7RE 16007391 Ki > 10000 nM T85943 D0S7HM 16041424 IC50 = 10 nM T85943 D0UF2N 21706 IC50 = 46000 nM T85943 D0VF6E 1401 IC50 = 20000 nM T85943 D0W3LI 153999 IC50 > 100000 nM T85943 D0XT0W 66555680 IC50 = 5900 nM T85943 D0Z4RC 24756910 IC50 = 11000 nM T85943 D03BNU 59604787 IC50 > 3500 nM T85943 D00PWQ 3820 IC50 = 15000 nM T85943 D01LMW 89899422 IC50 = 1423 nM T85943 D04SWX 56924694 IC50 = 399 nM T85943 D07FAF 53344793 IC50 > 10000 nM T85943 D0OE4F 4369496 IC50 = 7800 nM T85943 D0Y9PK 53346432 Ki > 20000 nM T85943 D01EFO 9864718 IC50 > 100000 nM T85943 D02YAQ 6603857 IC50 > 50000 nM T85943 D03QTP 1697 IC50 = 16000 nM T85943 D04FHB 6918852 Ki > 5000 nM T85943 D09HEV 6539952 IC50 = 42 nM T85943 D0F8DL 176155 IC50 = 5000 nM T85943 D0H8KG 5311382 IC50 = 9 nM T85943 D0HO1S 6711154 IC50 = 50000 nM T85943 D0IT6Q 3038522 IC50 = 30000 nM T85943 D0Q7HO 4705 IC50 = 1400 nM T85943 D0R2TM 5287736 IC50 > 10000 nM T85943 D0T3ME 156422 IC50 = 35000 nM T85943 C2BZ5G 1004 IC50 > 40000000 nM T85943 CB1VW3 1400 IC50 = 5 nM T85943 CK0GV2 2115 IC50 = 1000000 nM T85943 CZM9B7 2404 IC50 > 100000 nM T85943 CH21PG 2428 IC50 > 50000 nM T85943 CBPM40 4878 IC50 = 0.5 nM T85943 C97TNH 10177 IC50 = 18000 nM T85943 CG3YN1 10215 IC50 = 28000 nM T85943 CBE46X 14003 IC50 = 9000 nM T85943 CFA4M1 40320 Ki > 10000 nM T85943 CV96XE 83133 IC50 = 1000000 nM T85943 CDX60S 83430 IC50 = 4000000 nM T85943 C63WLY 89644 IC50 = 2.4 ug.mL-1 T85943 CK4I5X 100641 IC50 = 30900 nM T85943 C5JE2Z 104860 IC50 = 2.1 ug.mL-1 T85943 C3DY1O 122271 IC50 = 600000 nM T85943 C6Y9CV 151193 IC50 > 10000 nM T85943 CS5M0U 156118 IC50 = 35800 nM T85943 CA5CO8 157820 IC50 > 50000 nM T85943 CI1NA5 159926 IC50 > 10 ug.mL-1 T85943 CYBA43 177458 IC50 = 1.8 ug.mL-1 T85943 C30UNK 247352 IC50 = 3600 nM T85943 CWGJ94 256524 Ki = 18000 nM T85943 C9WA8F 341040 IC50 > 100000 nM T85943 CV3XI1 354479 IC50 = 158.49 nM T85943 CNP3M1 403661 IC50 = 2200 nM T85943 CC2R6G 409975 IC50 > 100000 nM T85943 CK0L4O 442514 IC50 = 440 nM T85943 C49LTY 444589 IC50 = 1800 nM T85943 C4MNG8 445840 IC50 > 5000 nM T85943 CH5A6J 446022 IC50 = 12700 nM T85943 CIE63B 446044 IC50 > 200000 nM T85943 C5JZD3 447520 IC50 = 3 nM T85943 CG1Y9D 447844 IC50 = 5900 nM T85943 CT6A4Y 448585 IC50 = 7000 nM T85943 C75EDQ 644355 IC50 > 30000 nM T85943 C5HPF3 644356 IC50 > 30000 nM T85943 CLV7T4 685639 Ki = 464 nM T85943 C9U7NK 1128774 IC50 > 100000 nM T85943 CQR4S9 1327207 Ki = 217 nM T85943 CYX87J 1474860 IC50 = 250 nM T85943 C6PTI2 2192320 Ki = 718 nM T85943 C4KZ1A 2363161 Ki = 900 nM T85943 CV7Y5T 2807058 IC50 > 100000 nM T85943 C2AFE3 2808988 IC50 = 253 nM T85943 CJBX04 3039851 IC50 > 100000 nM T85943 CCN9D5 3142817 IC50 = 190 nM T85943 C6LO1V 3320545 Ki = 200 nM T85943 CCFI27 3320547 Ki = 354 nM T85943 C0R5MH 3373694 IC50 = 190000 nM T85943 CC79BS 3448811 Ki = 522 nM T85943 C3JTC0 3643794 Ki = 221 nM T85943 CU5B1Z 4369491 IC50 > 50000 nM T85943 C9Y7IC 4390766 Ki = 64 nM T85943 CR5I7G 4573026 Ki = 569 nM T85943 CM5VN6 4600415 IC50 > 100000 nM T85943 CN7MT6 4750207 IC50 = 10000 nM T85943 CE74CV 5059890 IC50 > 1000 nM T85943 C97JHC 5157299 Ki = 1137 nM T85943 C8IAR2 5281657 IC50 = 35000 nM T85943 CN10FM 5281793 IC50 = 36200 nM T85943 CI68PW 5283685 IC50 = 2170 nM T85943 CXK0S6 5283727 IC50 = 1910 nM T85943 C6UL3A 5327821 IC50 = 6000 nM T85943 CR3OF4 5327822 IC50 = 6000 nM T85943 C9QMX2 5327823 IC50 = 75000 nM T85943 CA4G1B 5327824 IC50 = 2250 nM T85943 CY2NC3 5327825 IC50 = 5300 nM T85943 CDT07K 5327826 IC50 > 10000 nM T85943 CG36XB 5327827 IC50 = 8080 nM T85943 CF3Y6G 5327828 IC50 > 10000 nM T85943 CY1Z9E 5327829 IC50 = 400 nM T85943 CI51CH 5327830 IC50 = 7800 nM T85943 CUAW78 5327831 IC50 = 220 nM T85943 CC9US2 5327832 IC50 > 10000 nM T85943 CVGK98 5327833 IC50 = 2400 nM T85943 CGWP86 5327834 IC50 > 10000 nM T85943 C10RVD 5327835 IC50 > 10000 nM T85943 CD6B2A 5327836 IC50 = 2090 nM T85943 CY1O6K 5327837 IC50 > 10000 nM T85943 C1K8CJ 5327838 IC50 > 10000 nM T85943 CP15JO 5327839 IC50 > 10000 nM T85943 CWT9S8 5327840 IC50 = 2 nM T85943 C5EWD2 5327841 IC50 > 10000 nM T85943 C67JVQ 5327843 IC50 = 9800 nM T85943 CY23QP 5327844 IC50 > 10000 nM T85943 CN1X4Z 5327845 IC50 = 9800 nM T85943 C6TGI1 5327846 IC50 = 4900 nM T85943 CEMR07 5327847 IC50 > 10000 nM T85943 CB90GI 5327848 IC50 > 10000 nM T85943 CMC76E 5327864 IC50 = 260 nM T85943 C4ZW0Q 5327868 IC50 = 750 nM T85943 CI96EG 5327876 IC50 = 960 nM T85943 CT86OE 5327877 IC50 = 530 nM T85943 C23EZX 5327878 IC50 = 150 nM T85943 C63SAG 5327879 IC50 = 70 nM T85943 CT94BD 5327880 IC50 = 60 nM T85943 C3P8CG 5327885 IC50 = 16 nM T85943 CYRW80 5327889 IC50 = 10 nM T85943 C52MYD 5327893 IC50 = 492 nM T85943 CDA78E 5327896 IC50 = 20 nM T85943 CQ0ZP3 5327897 IC50 = 43 nM T85943 C7KIT4 5327898 IC50 = 223 nM T85943 CLH9Y3 5327908 IC50 = 17 nM T85943 CA7U3O 5327914 IC50 = 10 nM T85943 CQ54BE 5327946 IC50 > 12500 nM T85943 CCZ96X 5328096 IC50 = 6700 nM T85943 CW4XA5 5328097 IC50 = 600 nM T85943 CPT61U 5328112 IC50 = 220 nM T85943 CMW3F8 5328113 IC50 = 210 nM T85943 CXR9K1 5328115 IC50 = 73 nM T85943 CM0H5O 5328117 IC50 = 110 nM T85943 C7UJH5 5328121 IC50 = 210 nM T85943 CDM98R 5328125 IC50 > 50000 nM T85943 CDH5C1 5328126 IC50 > 50000 nM T85943 CDY2O3 5328134 IC50 = 23 nM T85943 CC1O0M 5328135 IC50 = 44 nM T85943 COT45A 5328149 IC50 = 31 nM T85943 CDV19S 5328354 IC50 > 50000 nM T85943 C1D0YT 5328357 IC50 > 50000 nM T85943 CC4O6Y 5328360 IC50 > 50000 nM T85943 C0Z8KJ 5328458 IC50 > 50000 nM T85943 C8C0RL 5328498 IC50 > 50000 nM T85943 CGW0I4 5328499 IC50 > 50000 nM T85943 CO4W7V 5328500 IC50 > 50000 nM T85943 CI5E6B 5328501 IC50 > 50000 nM T85943 CB3J1O 5328502 IC50 = 25000 nM T85943 CH2F1N 5328503 IC50 = 50000 nM T85943 C4AUK6 5328504 IC50 > 50000 nM T85943 CFSN21 5328505 IC50 > 50000 nM T85943 CWQO83 5328506 IC50 = 28000 nM T85943 CG5M7U 5328507 IC50 = 14000 nM T85943 C4FE0B 5328508 IC50 = 50000 nM T85943 CJM61R 5328509 IC50 = 50000 nM T85943 CIY48D 5328510 IC50 = 50000 nM T85943 CM3D5O 5328511 IC50 = 25000 nM T85943 CN8IE6 5328513 IC50 > 50000 nM T85943 C1XMV2 5328514 IC50 > 50000 nM T85943 CKEY79 5328515 IC50 > 50000 nM T85943 CT65IH 5328516 IC50 > 50000 nM T85943 CA18OW 5328517 IC50 = 460 nM T85943 CJX18A 5328518 IC50 = 40000 nM T85943 CI1BS6 5328519 IC50 > 50000 nM T85943 C2W7DN 5328520 IC50 > 50000 nM T85943 CDL94I 5328521 IC50 > 50000 nM T85943 CO04IH 5328522 IC50 > 50000 nM T85943 C7HPN8 5328523 IC50 > 50000 nM T85943 CPZD13 5328524 IC50 > 50000 nM T85943 C1M2CY 5328525 IC50 = 40000 nM T85943 CS3CR5 5328526 IC50 = 50000 nM T85943 CM9EJ7 5328527 IC50 > 50000 nM T85943 CJE94R 5328528 IC50 > 50000 nM T85943 C2NE5X 5328529 IC50 > 50000 nM T85943 CXR8Z6 5328530 IC50 > 50000 nM T85943 CQH57F 5328531 IC50 = 33500 nM T85943 C0MW1I 5328532 IC50 = 33300 nM T85943 CFWZ98 5328533 IC50 = 50000 nM T85943 CK4L8D 5328534 IC50 > 50000 nM T85943 C3UAX9 5328558 IC50 = 5100 nM T85943 C3NC0W 5328560 IC50 = 3500 nM T85943 CB9UI5 5328569 IC50 = 3800 nM T85943 CVEY01 5328570 IC50 = 2500 nM T85943 C64XYH 5328573 IC50 = 1500 nM T85943 CBE9M4 5328574 IC50 = 750 nM T85943 C5QE9H 5328575 IC50 = 2900 nM T85943 CE9PW4 5328576 IC50 = 1200 nM T85943 CJ78UZ 5328577 IC50 = 4400 nM T85943 C9S1MH 5328578 IC50 = 2900 nM T85943 CE62YD 5328579 IC50 = 1800 nM T85943 C72KTF 5328580 IC50 = 1500 nM T85943 CG38AH 5328581 IC50 = 100000 nM T85943 CGDE60 5328583 IC50 = 14000 nM T85943 COF98M 5328584 IC50 = 500 nM T85943 C23LDB 5328585 IC50 = 700 nM T85943 CA9PL4 5328588 IC50 = 1300 nM T85943 CQDX90 5328589 IC50 = 3200 nM T85943 CLZ2T7 5328590 IC50 = 2000 nM T85943 CMP24I 5328591 IC50 = 9300 nM T85943 C0TX2I 5328592 IC50 = 3200 nM T85943 C9JLN6 5328593 IC50 > 100000 nM T85943 C42LEK 5328594 IC50 > 100000 nM T85943 CVF12E 5328595 IC50 > 100000 nM T85943 CGN3C9 5328596 IC50 = 650 nM T85943 C91NOL 5328597 IC50 = 6000 nM T85943 C0PB9W 5328598 IC50 > 100000 nM T85943 C9P3LY 5328599 IC50 = 100000 nM T85943 CQNB13 5328600 IC50 > 100000 nM T85943 CK7IA1 5328601 IC50 > 100000 nM T85943 CNI91T 5328602 IC50 = 7700 nM T85943 C3AW9S 5328603 IC50 = 3900 nM T85943 CWEA08 5328604 IC50 = 5800 nM T85943 CCM96I 5328605 IC50 = 4500 nM T85943 C9NVC5 5328606 IC50 = 7200 nM T85943 CDX4Z7 5328607 IC50 > 100000 nM T85943 CB1S3D 5328608 IC50 = 100000 nM T85943 C7WL3M 5328609 IC50 = 3600 nM T85943 C69QIE 5328610 IC50 = 3500 nM T85943 C09SPY 5328611 IC50 = 5100 nM T85943 CO2CR8 5328612 IC50 > 100000 nM T85943 CR3W8H 5328613 IC50 > 100000 nM T85943 CB2HD4 5328614 IC50 = 3600 nM T85943 C5GWD8 5328615 IC50 = 11100 nM T85943 C0MU7G 5328616 IC50 > 50000 nM T85943 CH1X6G 5328617 IC50 = 5200 nM T85943 CR02JQ 5328618 IC50 = 9700 nM T85943 CP8G4Z 5328619 IC50 > 100000 nM T85943 C8YS2H 5328620 IC50 = 30700 nM T85943 CM80FN 5328621 IC50 > 50000 nM T85943 C16JYR 5328622 IC50 > 50000 nM T85943 CL6QD5 5328623 IC50 > 100000 nM T85943 CFB26C 5328624 IC50 > 100000 nM T85943 CDYX05 5328651 IC50 = 1000 nM T85943 C9T8XO 5328652 IC50 = 900 nM T85943 CQ0J3T 5328653 IC50 = 4100 nM T85943 CG2E4F 5328654 IC50 = 11000 nM T85943 CK91OW 5328655 IC50 = 5400 nM T85943 CQ1XL2 5328656 IC50 = 21000 nM T85943 C6M9VU 5328657 IC50 = 900 nM T85943 CNB05S 5328658 IC50 = 61000 nM T85943 C9HT4W 5328659 IC50 = 1300 nM T85943 C2VLD0 5328660 IC50 = 197000 nM T85943 C2NK7Y 5328661 IC50 = 2000 nM T85943 CI4M2B 5328662 IC50 = 7200 nM T85943 C2WO6V 5328663 IC50 = 1500 nM T85943 CDZL85 5328664 IC50 = 800 nM T85943 CUI4E1 5328665 IC50 = 600 nM T85943 C8WV3X 5328666 IC50 = 7000 nM T85943 CXG98R 5328667 IC50 = 2000 nM T85943 C78KGZ 5328668 IC50 = 4000 nM T85943 CIW52M 5328669 IC50 = 900 nM T85943 CVBE63 5328670 IC50 = 8000 nM T85943 CI0HM4 5328671 IC50 = 500 nM T85943 CLQ9F1 5328672 IC50 = 400 nM T85943 C16VPK 5328673 IC50 = 900 nM T85943 C3Y6RS 5328674 IC50 = 9000 nM T85943 CFS94T 5328675 IC50 = 900 nM T85943 CA6H5G 5328676 IC50 = 3400 nM T85943 C97DXG 5328677 IC50 = 1700 nM T85943 CDL1K2 5328678 IC50 = 600 nM T85943 CQ5PU7 5328679 IC50 = 1400 nM T85943 CWQ38R 5328680 IC50 = 600 nM T85943 C4N1QV 5328681 IC50 = 500 nM T85943 CA75QE 5328682 IC50 = 600 nM T85943 C7LJ9A 5328683 IC50 = 700 nM T85943 CE8Z9D 5328684 IC50 = 2000 nM T85943 CC1Y6B 5328685 IC50 = 700 nM T85943 C2A3IS 5328686 IC50 = 12000 nM T85943 CX35KY 5328687 IC50 = 400 nM T85943 CLP59M 5328688 IC50 = 9000 nM T85943 CXZE51 5328689 IC50 = 400 nM T85943 C4Q8ZX 5328690 IC50 = 24000 nM T85943 CA6BP0 5328691 IC50 = 15000 nM T85943 CPYH83 5328692 IC50 = 7700 nM T85943 C40AVM 5328693 IC50 = 14000 nM T85943 CFZ65W 5328694 IC50 = 12000 nM T85943 CUE30V 5328700 IC50 = 350 nM T85943 C9IH8T 5328701 IC50 = 420 nM T85943 CL61RQ 5328702 IC50 > 50000 nM T85943 C9T8GP 5328703 IC50 = 13000 nM T85943 CI9B1T 5328704 IC50 = 300 nM T85943 C8VEP0 5328705 IC50 = 44 nM T85943 C4QZ1J 5328706 IC50 = 24 nM T85943 CR0UB3 5328707 IC50 = 59 nM T85943 C4GCM3 5328708 IC50 = 41 nM T85943 CFG6I9 5328709 IC50 = 35 nM T85943 CY12MK 5328710 IC50 = 200 nM T85943 C13KGU 5328711 IC50 = 45 nM T85943 C7XN8T 5328712 IC50 = 540 nM T85943 CFK34R 5328713 IC50 = 790 nM T85943 C37VOE 5328714 IC50 = 550 nM T85943 CBH91D 5328715 IC50 = 1800 nM T85943 COL47I 5328716 IC50 = 78 nM T85943 COI8H6 5328717 IC50 = 32 nM T85943 C8UK0W 5328718 IC50 = 16 nM T85943 CO1EU7 5328719 IC50 = 28 nM T85943 CX9D7E 5328720 IC50 = 23 nM T85943 CR4VJ8 5328721 IC50 = 250 nM T85943 CTV12Y 5328722 IC50 = 1000 nM T85943 C50CGB 5328723 IC50 = 42 nM T85943 CEW4B8 5328724 IC50 = 110 nM T85943 CCKV98 5328725 IC50 = 11 nM T85943 CN9ST1 5328726 IC50 > 50000 nM T85943 CDZF47 5328727 IC50 > 50000 nM T85943 CZN6F4 5328728 IC50 > 50000 nM T85943 CKD93O 5328729 IC50 > 50000 nM T85943 C5ICG9 5328730 IC50 > 50000 nM T85943 CM25VZ 5328731 IC50 = 29000 nM T85943 C56SHL 5328732 IC50 > 50000 nM T85943 CPL1U9 5328734 IC50 = 14 nM T85943 CXH6C3 5328843 IC50 = 950 nM T85943 C0G6RT 5328852 IC50 = 53 nM T85943 C76ORW 5328887 IC50 = 30 nM T85943 CZ52SN 5328888 IC50 = 84 nM T85943 C07WIM 5328890 IC50 = 2200 nM T85943 CMB23Y 5328893 IC50 = 250 nM T85943 C13XBR 5328894 IC50 = 1200 nM T85943 CUP95N 5328895 IC50 = 320 nM T85943 C3FBS2 5328896 IC50 = 200 nM T85943 C6L4KS 5328898 IC50 = 11 nM T85943 CU7P9B 5328899 IC50 = 160 nM T85943 C48NEY 5328900 IC50 = 95 nM T85943 CJ9S8V 5328901 IC50 = 53 nM T85943 CY1M6A 5328902 IC50 = 90 nM T85943 CF09YD 5328903 IC50 = 40 nM T85943 CE18LC 5328904 IC50 = 61 nM T85943 CWAR54 5328905 IC50 = 1100 nM T85943 CWB31P 5328906 IC50 = 57 nM T85943 CDCZ21 5328907 IC50 = 10 nM T85943 C71RTK 5328908 IC50 = 6.2 nM T85943 C58CDW 5328909 IC50 = 95 nM T85943 C4FRB9 5328910 IC50 = 15 nM T85943 CS6L2C 5328911 IC50 = 19 nM T85943 C16ECF 5328912 IC50 = 220 nM T85943 C23VOL 5328913 IC50 = 3.8 nM T85943 C8LGK5 5328914 IC50 = 8.7 nM T85943 CH83QU 5328915 IC50 = 3.5 nM T85943 C8THL2 5328916 IC50 = 10 nM T85943 CPHM29 5328917 IC50 = 4.3 nM T85943 C2TH6S 5328918 IC50 = 1200 nM T85943 CXM58D 5328919 IC50 > 5000 nM T85943 C2F3OZ 5328920 IC50 = 190 nM T85943 CQ49ZV 5328921 IC50 = 66 nM T85943 CI2H1F 5328922 IC50 = 3 nM T85943 CN9RK8 5328923 IC50 = 4 nM T85943 C5Y1JL 5328924 IC50 = 120 nM T85943 CE6B1P 5328925 IC50 = 2.9 nM T85943 CMT12B 5328926 IC50 > 5000 nM T85943 C2GD3C 5328927 IC50 = 4.6 nM T85943 CA7JL3 5328928 IC50 = 390 nM T85943 CN17GS 5328929 IC50 = 81 nM T85943 CBJE74 5328930 IC50 = 1.6 nM T85943 C8BH9X 5328931 IC50 = 0.8 nM T85943 C34CIY 5328932 IC50 = 0.95 nM T85943 CWM79C 5328933 IC50 = 1.2 nM T85943 C7Y8HT 5328934 IC50 = 1.7 nM T85943 CSQ3Y9 5328935 IC50 = 1.1 nM T85943 CAW5X6 5328936 IC50 = 28 nM T85943 C89PYI 5328937 IC50 = 2.3 nM T85943 CK0BG7 5328938 IC50 = 1.3 nM T85943 C3J5TO 5328939 IC50 = 2.5 nM T85943 CK7HC3 5328941 IC50 = 0.77 nM T85943 C53MGP 5328943 IC50 = 1.1 nM T85943 CCZ48B 5328944 IC50 = 1.1 nM T85943 C17WBH 5328945 IC50 = 0.76 nM T85943 C3GJ5F 5328946 IC50 = 1.4 nM T85943 C6JN2W 5328947 IC50 = 1.2 nM T85943 C8NW2G 5328948 IC50 = 0.64 nM T85943 CZAP80 5328949 IC50 = 9.3 nM T85943 CW1Z4M 5328950 IC50 = 1.9 nM T85943 CG6IA5 5328951 IC50 = 2.1 nM T85943 C02PBT 5328952 IC50 = 3 nM T85943 CU3A7R 5328953 IC50 = 2.3 nM T85943 C5R9DV 5328990 IC50 = 17000 nM T85943 CDNP54 5328991 IC50 = 5100 nM T85943 C6J5YD 5328992 IC50 = 4400 nM T85943 CY5L7F 5328993 IC50 = 680 nM T85943 CCV0B4 5328994 IC50 = 100 nM T85943 C3A1ER 5328995 IC50 = 170 nM T85943 CA05KW 5328996 IC50 > 50000 nM T85943 CF0PG3 5328997 IC50 > 50000 nM T85943 C68UKW 5328998 IC50 > 50000 nM T85943 CU4XT5 5328999 IC50 > 50000 nM T85943 CPK58V 5329000 IC50 > 50000 nM T85943 C10WHP 5329001 IC50 = 3800 nM T85943 C7HB6C 5329002 IC50 > 50000 nM T85943 C5D4WA 5329003 IC50 > 50000 nM T85943 CWX63A 5329004 IC50 > 50000 nM T85943 CSY10K 5329111 IC50 = 19330 nM T85943 CV7FG2 5329112 IC50 = 4410 nM T85943 C4VQ2R 5329113 IC50 = 1410 nM T85943 C2SQL0 5329114 IC50 = 210 nM T85943 CNI13Q 5329115 IC50 = 800 nM T85943 C1JF3N 5329116 IC50 = 1350 nM T85943 C19GHD 5329117 IC50 > 50000 nM T85943 C6C8RV 5329118 IC50 = 410 nM T85943 C5V8FR 5329119 IC50 = 17500 nM T85943 CYU89T 5329120 IC50 = 4170 nM T85943 CDU9H6 5329121 IC50 > 50000 nM T85943 CMAV05 5329122 IC50 = 360 nM T85943 CG8B3E 5329123 IC50 > 50000 nM T85943 CW5U4J 5329124 IC50 = 1650 nM T85943 C39FIH 5329125 IC50 = 10430 nM T85943 CMY9D6 5329126 IC50 > 50000 nM T85943 C6VO5Z 5329127 IC50 = 10430 nM T85943 CM7B2T 5329128 IC50 = 36400 nM T85943 C9GXO6 5329129 IC50 > 50000 nM T85943 CP5AI7 5329130 IC50 > 50000 nM T85943 C4I3ZO 5329131 IC50 > 50000 nM T85943 C8IF1G 5329132 IC50 > 50000 nM T85943 CE68LC 5329133 IC50 > 50000 nM T85943 CGWD98 5329154 IC50 = 4740 nM T85943 C4PD0K 5329156 IC50 = 80 nM T85943 C0RWT8 5329157 IC50 = 120 nM T85943 C3MU5S 5329158 IC50 > 20000 nM T85943 CN6O4R 5329159 IC50 > 20000 nM T85943 CG68DI 5329160 IC50 > 20000 nM T85943 CYR7V0 5329161 IC50 > 20000 nM T85943 C9BXE2 5329162 IC50 > 20000 nM T85943 CY4V5Z 5329163 IC50 = 1890 nM T85943 CI64YA 5329164 IC50 = 1270 nM T85943 C2ZV0O 5329165 IC50 = 680 nM T85943 CAB53L 5329166 IC50 = 60 nM T85943 CTW9R8 5329167 IC50 = 1390 nM T85943 C8A3TJ 5329168 IC50 = 110 nM T85943 CVTD82 5329169 IC50 = 100 nM T85943 CQ5WK1 5329170 IC50 = 840 nM T85943 CNC9T7 5329171 IC50 = 60 nM T85943 CUE64R 5329179 IC50 = 292000 nM T85943 CHA68G 5329180 IC50 = 96000 nM T85943 CNTD47 5329181 IC50 = 205000 nM T85943 CYFD81 5329182 IC50 = 259000 nM T85943 C21IKR 5329183 IC50 > 500000 nM T85943 C45ZME 5329185 IC50 = 135000 nM T85943 C5U7DB 5329186 IC50 = 156000 nM T85943 CQ6X8M 5329189 IC50 = 115000 nM T85943 C5HG9S 5329194 IC50 = 39000 nM T85943 CHV5Y6 5329195 IC50 = 45000 nM T85943 C3DOZ9 5329196 IC50 = 50000 nM T85943 CT61MB 5329197 IC50 = 40000 nM T85943 C6OT4G 5329198 IC50 = 489000 nM T85943 CROF47 5329199 IC50 > 500000 nM T85943 CHNM67 5329200 IC50 > 500000 nM T85943 C1G6ZU 5329201 IC50 > 500000 nM T85943 CA2HW9 5329202 IC50 = 92000 nM T85943 C30CUW 5329203 IC50 = 98000 nM T85943 C0UY4Q 5329204 IC50 = 149000 nM T85943 C3QIN5 5329205 IC50 = 132000 nM T85943 C5OBU1 5329206 IC50 = 32000 nM T85943 C2GKT3 5329207 IC50 = 37000 nM T85943 CKB23P 5329209 IC50 = 143000 nM T85943 CDL19N 5329212 IC50 = 49000 nM T85943 CI03PS 5329214 IC50 = 72000 nM T85943 C43NAT 5329215 IC50 = 206000 nM T85943 C9D3WP 5329216 IC50 = 274000 nM T85943 CS2I1H 5329217 IC50 = 72000 nM T85943 CQ70YG 5329218 IC50 = 64000 nM T85943 C6OL3X 5329220 IC50 = 75000 nM T85943 C2J4ZO 5329221 IC50 = 99000 nM T85943 CO87DJ 5329222 IC50 = 282000 nM T85943 C5LW1G 5329223 IC50 = 95000 nM T85943 CRB3S4 5329224 IC50 = 78000 nM T85943 CU68QR 5329225 IC50 = 60000 nM T85943 C4P7QH 5329226 IC50 = 161000 nM T85943 CWF7K8 5329227 IC50 = 35000 nM T85943 CJ6VE0 5329228 IC50 = 68000 nM T85943 C4RUV5 5329453 IC50 = 50 nM T85943 C73DUO 5330057 IC50 = 34 nM T85943 C9EM4B 5330058 IC50 = 13 nM T85943 C65GIE 5330059 IC50 = 630 nM T85943 CVUZ92 5330060 IC50 = 7.2 nM T85943 CVSA95 5330061 IC50 = 7.4 nM T85943 C2FVK5 5330062 IC50 = 17 nM T85943 CY9J7I 5330063 IC50 = 52 nM T85943 C5A0RM 5330064 IC50 = 9.1 nM T85943 C6VY7I 5330065 IC50 = 890 nM T85943 C9IX4U 5330066 IC50 = 13 nM T85943 CS2AW3 5330067 IC50 = 1400 nM T85943 CX1P8Q 5330068 IC50 = 110 nM T85943 CX68VG 5330069 IC50 = 8.8 nM T85943 C2KBS0 5330070 IC50 = 15 nM T85943 CZMK91 5330071 IC50 = 50 nM T85943 C2O6JM 5330072 IC50 = 980 nM T85943 CLVI54 5330073 IC50 = 140 nM T85943 CD1NL0 5330074 IC50 = 53 nM T85943 C2CZJ1 5330075 IC50 = 430 nM T85943 CLZ2W6 5330076 IC50 = 67 nM T85943 C6TXZ5 5330077 IC50 = 1300 nM T85943 CX0GQ4 5330078 IC50 = 690 nM T85943 CEHP64 5330079 IC50 = 25 nM T85943 CN93OL 5330080 IC50 = 420 nM T85943 CXLB39 5330081 IC50 = 2 nM T85943 CUOM76 5330082 IC50 = 2.4 nM T85943 CHZ3F9 5330083 IC50 = 1.4 nM T85943 CF58NA 5330084 IC50 = 230 nM T85943 C1F5NT 5330085 IC50 = 87 nM T85943 CE80MZ 5330086 IC50 = 9 nM T85943 CQPB30 5330087 IC50 = 6.6 nM T85943 CVA4J7 5330088 IC50 = 8.3 nM T85943 C7CXF8 5330089 IC50 = 12 nM T85943 CTIR20 5330090 IC50 = 24 nM T85943 C04MYD 5330091 IC50 = 63 nM T85943 C0JUX8 5330092 IC50 = 13 nM T85943 CKX46W 5330093 IC50 = 1400 nM T85943 CU17ND 5330094 IC50 = 2.7 nM T85943 CZ7JV0 5330095 IC50 = 2.5 nM T85943 C1LSN5 5330096 IC50 = 5.7 nM T85943 CZ9FL0 5330097 IC50 = 440 nM T85943 CSLB59 5330098 IC50 = 240 nM T85943 CM98RH 5330099 IC50 = 3.8 nM T85943 CR79PF 5330100 IC50 = 1.4 nM T85943 C0RSM4 5330101 IC50 = 2.3 nM T85943 CTZ9F6 5330105 IC50 = 280 nM T85943 CIQ58M 5330106 IC50 = 5.1 nM T85943 CQ5I4P 5330107 IC50 = 2.8 nM T85943 CS60BJ 5330108 IC50 = 12 nM T85943 C5YMA2 5330109 IC50 = 25 nM T85943 C1WZH8 5330110 IC50 = 1.5 nM T85943 C7NP4A 5330111 IC50 = 4.7 nM T85943 C7CA8T 5330112 IC50 = 14 nM T85943 CB0QZ2 5330117 IC50 = 180 nM T85943 C7QZL3 5330118 IC50 = 67 nM T85943 CNR9B8 5330119 IC50 = 620 nM T85943 CXY2I9 5330120 IC50 = 43 nM T85943 CDF96J 5330121 IC50 = 120 nM T85943 C7BPR2 5330122 IC50 = 29 nM T85943 CC4ZJ3 5330123 IC50 = 9 nM T85943 CLV0T6 5330124 IC50 = 200 nM T85943 CY7K6I 5330170 IC50 = 37 nM T85943 CSNZ07 5330171 IC50 = 560 nM T85943 C1KY4Q 5330172 IC50 = 477 nM T85943 CI32HV 5330173 IC50 = 10 nM T85943 CI4K3U 5330174 IC50 = 963 nM T85943 C7Y2VN 5330175 IC50 = 5 nM T85943 C3Q1SK 5330176 IC50 = 16 nM T85943 CC4Z9K 5330178 IC50 = 10 nM T85943 C2H1EQ 5330179 IC50 = 30 nM T85943 C04DHT 5330180 IC50 = 10 nM T85943 C54GDC 5330181 IC50 = 433 nM T85943 COF57G 5330182 IC50 < 4 nM T85943 CU9YJ1 5330183 IC50 = 177 nM T85943 CH9SZ3 5330184 IC50 = 40 nM T85943 CW3JY1 5330185 IC50 = 260 nM T85943 CA09XJ 5330186 IC50 = 380 nM T85943 CA5H0W 5330187 IC50 = 14 nM T85943 C5RK3H 5330188 IC50 < 4 nM T85943 C6NMP8 5330189 IC50 < 4 nM T85943 CW81JE 5330190 IC50 = 300 nM T85943 CL3KH1 5330191 IC50 = 270 nM T85943 C6A4WQ 5330192 IC50 = 760 nM T85943 CWF2G1 5330193 IC50 = 370 nM T85943 CQDI38 5330194 IC50 = 10 nM T85943 CUZ0I1 5330195 IC50 = 50 nM T85943 CD7U5B 5330196 IC50 = 5 nM T85943 CB23PA 5330197 IC50 < 4 nM T85943 C6BPR5 5330198 IC50 = 90 nM T85943 C5PL8M 5330199 IC50 = 21000 nM T85943 C94SHE 5330408 IC50 = 2500 nM T85943 C06CQH 5330409 IC50 = 250 nM T85943 C4S0FN 5330411 IC50 = 21 nM T85943 CA7R2B 5330413 IC50 > 10000 nM T85943 CK9SC1 5330414 IC50 = 830 nM T85943 CUN0I9 5330415 IC50 = 580 nM T85943 CVI1M2 5330419 IC50 = 56 nM T85943 C5SY4O 5330420 IC50 = 13 nM T85943 C95JFX 5330421 IC50 = 51 nM T85943 C7Y6KO 5330422 IC50 = 300 nM T85943 CM1U2R 5330423 IC50 = 13 nM T85943 C0V3LI 5330424 IC50 = 14 nM T85943 C7WOR4 5330425 IC50 = 47 nM T85943 CFKG51 5330426 IC50 = 2.1 nM T85943 C3C7JY 5330427 IC50 = 1.5 nM T85943 CT29GB 5330428 IC50 = 1.8 nM T85943 CLT49W 5330429 IC50 = 1.1 nM T85943 CIFU48 5330430 IC50 = 2.1 nM T85943 CYLX01 5330431 IC50 = 110 nM T85943 CD7CS0 5330432 IC50 = 2.6 nM T85943 CIZO27 5330433 IC50 = 1.2 nM T85943 CC24DW 5330434 IC50 = 13 nM T85943 CE7MG9 5330435 IC50 = 0.15 nM T85943 CXJ15Q 5330436 IC50 = 42 nM T85943 CUEZ35 5330437 IC50 = 37 nM T85943 CR25PZ 5330438 IC50 = 61 nM T85943 CUY6J4 5330439 IC50 = 0.72 nM T85943 C67SJG 5330440 IC50 = 19 nM T85943 CWV8E5 5330441 IC50 = 0.55 nM T85943 CQ4F5A 5330442 IC50 = 0.48 nM T85943 CY4CV0 5330443 IC50 = 210 nM T85943 C20OMA 5330444 IC50 = 0.69 nM T85943 CWZV82 5330445 IC50 = 50 nM T85943 CM7NA3 5330446 IC50 = 2 nM T85943 C9DH1B 5330447 IC50 = 150 nM T85943 C9Z0RF 5330448 IC50 = 15 nM T85943 C7QN8J 5330449 IC50 = 7 nM T85943 C6TPJ0 5330450 IC50 = 74 nM T85943 CA7BN5 5330451 IC50 = 11 nM T85943 C1WS3I 5330452 IC50 = 28 nM T85943 C94GRU 5330453 IC50 = 3.3 nM T85943 CYL2I4 5330454 IC50 = 3 nM T85943 C8WF6N 5330455 IC50 = 29 nM T85943 CR0O9Q 5330456 IC50 = 14 nM T85943 C67HIU 5330457 IC50 = 3.7 nM T85943 CSM0H3 5330458 IC50 = 14 nM T85943 CH2JS0 5330459 IC50 = 3.8 nM T85943 CK51NU 5330460 IC50 = 4.7 nM T85943 CMK0B9 5330461 IC50 = 4000 nM T85943 CO9YW2 5330463 IC50 = 340 nM T85943 CP7OD5 5330464 IC50 = 490 nM T85943 C6BI3U 5330465 IC50 = 830 nM T85943 CH83MG 5330466 IC50 = 2700 nM T85943 CIC0K3 5330467 IC50 = 5200 nM T85943 CC2E4Q 5330468 IC50 = 190 nM T85943 CD7CV2 5330469 IC50 = 63 nM T85943 C9D8IH 5330470 IC50 = 110 nM T85943 C5NO9G 5330471 IC50 = 180 nM T85943 C6XWB5 5330472 IC50 = 980 nM T85943 CDK95L 5330473 IC50 = 470 nM T85943 CR8QY3 5330474 IC50 = 170 nM T85943 C1YWE0 5330475 IC50 = 200 nM T85943 CI5PU3 5330476 IC50 > 10000 nM T85943 CU2N5S 5330477 IC50 > 10000 nM T85943 C7E0IC 5330478 IC50 = 290 nM T85943 CL2F8W 5330480 IC50 = 4.2 nM T85943 CX0AJ4 5330481 IC50 = 9.9 nM T85943 CGNC60 5330482 IC50 = 42 nM T85943 CSUD39 5330483 IC50 = 12 nM T85943 C5B4LP 5330484 IC50 = 47 nM T85943 CZ92XS 5330485 IC50 = 16 nM T85943 C1YL0D 5330486 IC50 = 21 nM T85943 C5YO6P 5330487 IC50 = 46 nM T85943 CKQG53 5330488 IC50 = 19 nM T85943 CY58JU 5330489 IC50 = 89 nM T85943 CL1EK9 5330490 IC50 = 160 nM T85943 C82SHZ 5330491 IC50 = 17 nM T85943 CNH9S0 5330492 IC50 = 34 nM T85943 CN9U6A 5330493 IC50 = 610 nM T85943 C3AQK7 5330494 IC50 = 740 nM T85943 C3QMZ6 5330496 IC50 = 910 nM T85943 C8L5BP 5330501 IC50 = 4.2 nM T85943 C21DKT 5330502 IC50 = 0.6 nM T85943 CM8FS5 5330504 IC50 = 200 nM T85943 CUIE17 5330505 IC50 = 3100 nM T85943 C0LU2O 5330507 IC50 = 380 nM T85943 C05QNO 5330508 IC50 = 12000 nM T85943 COZ3C0 5330509 IC50 = 1600 nM T85943 CXE7Y4 5330510 IC50 = 97 nM T85943 CK89CN 5330511 IC50 = 180 nM T85943 CEN6U5 5330512 IC50 = 2300 nM T85943 CYGE90 5330513 IC50 = 320 nM T85943 C3XTC0 5330514 IC50 = 19 nM T85943 C08QVB 5330515 IC50 = 15 nM T85943 C4H5UW 5330516 IC50 = 320 nM T85943 CR8L2I 5330517 IC50 = 420 nM T85943 CU2D5W 5330518 IC50 = 530 nM T85943 CND78K 5330519 IC50 = 83 nM T85943 CGH4M9 5330520 IC50 = 440 nM T85943 CU63CT 5330521 IC50 = 65 nM T85943 C9DLK7 5330522 IC50 = 8.4 nM T85943 CJL2S7 5330523 IC50 = 57 nM T85943 C9NBG7 5330546 IC50 > 30000 nM T85943 CS3A8F 5331081 IC50 > 20000 nM T85943 CG4W8K 5331082 IC50 > 20000 nM T85943 CD4C2A 5331083 IC50 = 13000 nM T85943 C6AT8V 5331084 IC50 > 20000 nM T85943 CJVS23 5331085 IC50 > 20000 nM T85943 CZ29FN 5331086 IC50 > 20000 nM T85943 CYL78A 5331087 IC50 > 20000 nM T85943 CJ87XR 5331088 IC50 > 20000 nM T85943 CFB3K7 5331089 IC50 > 20000 nM T85943 C9WY1O 5331090 IC50 > 20000 nM T85943 C9ZK3D 5331091 IC50 > 20000 nM T85943 C6RJC8 5331092 IC50 = 1100 nM T85943 C0IOY8 5331093 IC50 > 20000 nM T85943 CMD08O 5331094 IC50 = 8400 nM T85943 CM47KI 5351344 IC50 > 10000 nM T85943 CDQ3M7 5359485 IC50 = 4.4 ug.mL-1 T85943 C54BYP 5360741 IC50 = 1.2 ug.mL-1 T85943 CDK3J0 5703619 IC50 = 7.9 nM T85943 C7WI1P 6326454 IC50 = 65000 nM T85943 CLB02J 6326455 IC50 = 66000 nM T85943 CZK47S 6326456 IC50 = 200000 nM T85943 CS23WK 6326457 IC50 = 31000 nM T85943 CR59JT 6326458 IC50 = 68000 nM T85943 CN1GO8 6326459 IC50 = 18000 nM T85943 CY4WT0 6326460 IC50 = 123000 nM T85943 CEW21T 6326461 IC50 = 130000 nM T85943 C3PNU9 6326462 IC50 = 87000 nM T85943 CLTQ35 6326463 IC50 = 62000 nM T85943 CU6S2L 6326464 IC50 = 72000 nM T85943 C61JMS 6419746 IC50 = 4400 nM T85943 C4RVA6 6440397 IC50 = 74000 nM T85943 CA31PJ 6539953 IC50 = 35 nM T85943 C64ZJA 6539954 IC50 = 65 nM T85943 CBD1H7 6539955 IC50 = 427 nM T85943 CWHY29 6539956 IC50 = 189 nM T85943 CW76RA 6539957 IC50 = 12.5 nM T85943 C7K1QS 6539958 IC50 = 310 nM T85943 CJ7IL2 6539959 IC50 = 3190 nM T85943 CAE95J 6539960 IC50 = 463 nM T85943 CH86XJ 6539961 IC50 = 68 nM T85943 C41FUH 6539962 IC50 = 155 nM T85943 C7M2JP 6539963 IC50 = 460 nM T85943 CS5V1C 6539964 IC50 = 115 nM T85943 C10FYS 6539966 IC50 = 43 nM T85943 CIS1T3 6539967 IC50 = 526 nM T85943 CP0XI6 6603792 IC50 = 560 nM T85943 CG17TN 6914611 IC50 = 2000 nM T85943 C7E2QK 6914613 IC50 > 50000 nM T85943 CO9N0D 7946867 Ki = 334 nM T85943 C4G9WR 9547398 IC50 > 100000 nM T85943 C76CUP 9547698 IC50 = 2240 nM T85943 C3R5VW 9547983 IC50 = 162 nM T85943 CIR12S 9564690 IC50 = 269 nM T85943 CIJ25V 9794947 IC50 > 5000000 nM T85943 CZR3M4 9799152 IC50 > 100000 nM T85943 CI80BK 9803350 IC50 = 60 nM T85943 CSM34J 9804627 IC50 = 298 nM T85943 CB9ZH4 9805421 IC50 = 38 nM T85943 CX5FE7 9811952 Ki = 700000 nM T85943 CI3O6X 9814609 IC50 > 100000 nM T85943 CUNV09 9816954 IC50 > 100000 nM T85943 CX9DG5 9822042 IC50 > 100000 nM T85943 C6QBF8 9823235 Ki = 333 nM T85943 C1E2DV 9826083 IC50 > 10000 nM T85943 C9TAL6 9826308 IC50 > 30000 nM T85943 C8J1OL 9826373 IC50 = 68000 nM T85943 CI50RX 9829289 IC50 = 2200 nM T85943 CCE7V5 9829458 IC50 = 26000 nM T85943 CSH0A9 9847014 IC50 = 500 nM T85943 CXQ9J0 9856983 Ki = 1062 nM T85943 C1QM0N 9858715 Ki = 1059 nM T85943 CP2HX8 9859520 IC50 = 4400000 nM T85943 C3UQL7 9860872 IC50 = 93000 nM T85943 CTN7L4 9869773 IC50 = 800 nM T85943 CM5Z8X 9869943 IC50 = 0.2 nM T85943 CG41CN 9870411 IC50 = 483000 nM T85943 CG75DM 9872400 IC50 = 2 nM T85943 C1W4JG 9872939 IC50 = 1000 nM T85943 CD1PK3 9873683 IC50 = 6900 nM T85943 CY70OD 9882602 IC50 > 100000 nM T85943 CV1A2S 9883384 IC50 > 10000 nM T85943 C9ER0N 9886767 IC50 = 141 nM T85943 C20NKA 9889351 IC50 > 100000 nM T85943 CI63ZK 9890528 IC50 = 2800 nM T85943 CHF7G5 9890746 IC50 > 30000 nM T85943 C10RSK 9895224 IC50 = 5300 nM T85943 CUG5J1 9901007 Ki = 181 nM T85943 C7UIP5 9901505 Ki = 1288 nM T85943 C3EUB4 9911005 IC50 > 30000 nM T85943 CYW49X 9927718 IC50 = 10 nM T85943 CPQ13K 9933545 IC50 = 3480000 nM T85943 CRK63X 9933645 Ki = 13 nM T85943 CTV25B 9934643 IC50 = 0.45 nM T85943 CH7U4A 9938211 IC50 = 8600 nM T85943 C41OBR 9939269 IC50 = 350 nM T85943 CIZ13L 9943193 IC50 = 16000 nM T85943 CUKH27 9943194 IC50 = 14000 nM T85943 CU78NO 9947433 IC50 = 9000 nM T85943 CZC4L7 9948194 IC50 = 199.53 nM T85943 CYI65J 9948215 IC50 > 100000 nM T85943 C54ZXH 9950678 IC50 = 610 nM T85943 CYT7R9 9953676 IC50 > 100000 nM T85943 CV34AB 9958125 IC50 > 100000 nM T85943 CJ40GO 9965429 IC50 > 100000 nM T85943 C75QCM 9969776 Ki = 277 nM T85943 CAH50Y 9970231 IC50 > 50000 nM T85943 CG8CU4 9970992 IC50 = 38000 nM T85943 CQ0SW7 9978312 IC50 = 13000 nM T85943 C84LCW 9985193 IC50 = 102000 nM T85943 C29SOH 9985870 IC50 = 5500 nM T85943 CCYJ69 9986663 IC50 = 7 nM T85943 C26QHZ 10005638 IC50 > 10000 nM T85943 CUY0F8 10005715 IC50 > 10000 nM T85943 CYX27A 10006987 IC50 = 35 nM T85943 C0EWK9 10007087 IC50 = 1000 nM T85943 C93XNT 10007694 IC50 = 41 nM T85943 CA0BL8 10008474 IC50 = 12500 nM T85943 C8UYB4 10008492 IC50 = 3 nM T85943 CH7DN2 10009462 IC50 = 4300 nM T85943 C7Q5CN 10015651 IC50 = 25000 nM T85943 CRY61O 10019770 IC50 = 3500 nM T85943 C53UTR 10022185 IC50 > 100000 nM T85943 CR8DA1 10024683 IC50 > 100000 nM T85943 CMZ2S8 10029735 IC50 = 341 nM T85943 CGD5O1 10030767 IC50 = 3500 nM T85943 C1O4GZ 10031003 IC50 = 54000 nM T85943 C19XDW 10032479 IC50 = 15600 nM T85943 C0IA4P 10037831 IC50 = 28800 nM T85943 CXL0R8 10038606 IC50 > 50000 nM T85943 C0G5DK 10039959 IC50 = 126000 nM T85943 C25JLD 10043994 IC50 = 64000 nM T85943 CLA93G 10047202 IC50 = 1480 nM T85943 C3LCH5 10047545 IC50 > 100000 nM T85943 C54AEL 10048519 IC50 > 100000 nM T85943 C5ZY0I 10050705 IC50 = 2.3 nM T85943 C9VQZ3 10053637 IC50 = 47000 nM T85943 CFS2H4 10053638 IC50 > 50000 nM T85943 CGHK50 10054795 IC50 = 150 nM T85943 CUJR40 10062694 EC50 = 13 nM T85943 C6K0XB 10064040 IC50 = 50000 nM T85943 CBF54I 10066030 IC50 = 1000 nM T85943 CU2KS9 10066538 IC50 = 13000 nM T85943 C2L3JB 10068026 IC50 = 28000 nM T85943 CEKL46 10070245 IC50 = 36 nM T85943 C2P6HN 10071040 IC50 = 234 nM T85943 C7J8YN 10073101 IC50 > 100000 nM T85943 CF1D6Y 10075240 IC50 > 10000 nM T85943 CTAY63 10076476 IC50 = 7300 nM T85943 CD5B6O 10076837 IC50 > 50000 nM T85943 CU2JO1 10081832 IC50 = 100000 nM T85943 C8A1TH 10085171 IC50 > 50000 nM T85943 CFDU07 10090006 Ki = 794.33 nM T85943 C8G5RH 10095463 IC50 = 150 nM T85943 CXL3W1 10096996 IC50 = 769000 nM T85943 CLYU17 10099175 IC50 = 7000 nM T85943 CM2VB6 10100735 IC50 = 7300 nM T85943 CK50LJ 10100761 IC50 = 3500 nM T85943 C67CZY 10102298 IC50 = 25000 nM T85943 C3P8WK 10110378 IC50 > 100000 nM T85943 C63CFD 10111108 IC50 > 100000 nM T85943 CV9B4X 10112611 Ki = 1735 nM T85943 CY28QV 10113430 IC50 = 30 nM T85943 C7TA9J 10113568 IC50 = 537.03 nM T85943 CLA2N6 10133600 Ki = 201 nM T85943 CKL3V4 10134576 Ki > 500 nM T85943 CL42XS 10136330 IC50 > 100000 nM T85943 CL25BM 10138376 IC50 = 2360 nM T85943 CUW34X 10157645 IC50 > 100000 nM T85943 CV73FD 10157920 Ki > 38 nM T85943 CQN8M3 10159519 Ki = 681 nM T85943 C5QHB6 10161543 IC50 = 1780 nM T85943 C7X6KB 10165834 IC50 < 4 nM T85943 C3KHT0 10179373 Ki = 720 nM T85943 CXD4Z2 10180161 Ki = 461 nM T85943 COC30E 10181160 IC50 > 100000 nM T85943 C67PWJ 10181898 IC50 = 10 nM T85943 CO08KZ 10182284 Ki > 3000 nM T85943 CHSX56 10186317 IC50 = 7 nM T85943 C7PEG0 10200408 Ki = 1258 nM T85943 C8B0CW 10207842 IC50 = 6 nM T85943 C0D3XA 10209627 IC50 < 4 nM T85943 C0R5AX 10215912 IC50 = 2377 nM T85943 CI8MW4 10216627 IC50 = 12100 nM T85943 CPE29J 10229538 IC50 < 4 nM T85943 CD7J3O 10231458 IC50 > 30000 nM T85943 C97GRN 10248747 IC50 = 12 nM T85943 C32KTH 10253992 IC50 = 500 nM T85943 CT9R2O 10255644 IC50 = 5.5 nM T85943 CG2TF7 10255849 IC50 = 8300 nM T85943 CBR9P3 10257058 IC50 = 15200 nM T85943 C2H1XP 10261645 IC50 = 385000 nM T85943 C6G8NR 10264200 IC50 > 50000 nM T85943 C3HF6S 10264201 IC50 > 50000 nM T85943 CF81EM 10265006 IC50 > 50000 nM T85943 CHFZ23 10266516 IC50 > 100000 nM T85943 CWY4U3 10267270 IC50 = 1.995 nM T85943 CGF6I3 10267834 Ki = 393 nM T85943 C28AEC 10268530 Ki = 800 nM T85943 C6DC8Q 10275163 IC50 = 100 nM T85943 CI34AB 10276115 IC50 = 5 nM T85943 CW8OB2 10279981 IC50 = 10 nM T85943 CGN04D 10288960 IC50 = 40 nM T85943 CF9N7Y 10292186 Ki > 1000 nM T85943 CN51JQ 10292737 IC50 = 46000 nM T85943 C8U5LM 10295900 IC50 = 18 nM T85943 C8RD3V 10301884 IC50 < 4 nM T85943 CAM42B 10301885 IC50 = 80 nM T85943 C1KFM8 10318154 IC50 > 100000 nM T85943 C27CDR 10319118 IC50 > 50000 nM T85943 C62MZJ 10320122 Ki = 700 nM T85943 C5CBF9 10320381 IC50 = 30 nM T85943 CAV1N3 10325005 IC50 = 8000 nM T85943 CCK42E 10327195 IC50 = 800 nM T85943 CX7NM0 10327196 IC50 = 5400 nM T85943 CQ03XB 10327197 IC50 = 4200 nM T85943 COC7P1 10333957 IC50 > 50000 nM T85943 CQ80HY 10337047 IC50 > 100000 nM T85943 CET21U 10337153 IC50 > 100000 nM T85943 CUN52O 10345191 IC50 = 18 nM T85943 CP4M1C 10347718 IC50 = 53000 nM T85943 CD2H0G 10347728 IC50 = 22500 nM T85943 CNJ97S 10348925 IC50 = 4000 nM T85943 C7XFS9 10349305 IC50 = 20000 nM T85943 CZ0UL8 10349829 IC50 = 2500 nM T85943 CYCM39 10355659 IC50 > 50000 nM T85943 C37AMD 10356450 IC50 > 50000 nM T85943 C4DOQ9 10356451 IC50 = 38400 nM T85943 C19VUI 10360971 IC50 > 100000 nM T85943 CDS29Z 10366675 IC50 = 43 nM T85943 C8H1OJ 10371203 IC50 = 8000 nM T85943 C6DH4W 10382627 IC50 = 410 nM T85943 C4NO1Y 10383878 Ki = 2511.89 nM T85943 CHN1P0 10384072 IC50 > 50000 nM T85943 C36GIL 10386874 IC50 = 800 nM T85943 CA8B5T 10390073 IC50 = 8000 nM T85943 COR4A9 10393855 IC50 = 200 nM T85943 CYX5T0 10394312 IC50 = 2000 nM T85943 C7Y4SQ 10394740 IC50 = 150 nM T85943 CPS79C 10402283 IC50 = 0.035 ug.mL-1 T85943 CL3NV7 10404115 IC50 = 1500 nM T85943 CF74ID 10406267 IC50 = 8000 nM T85943 C9RCU7 10408993 IC50 = 50000 nM T85943 C4PV3R 10409198 IC50 = 11500 nM T85943 C2VR3A 10410783 IC50 = 2500 nM T85943 CQBD84 10410849 IC50 > 50000 nM T85943 CLAX64 10413508 IC50 = 200 nM T85943 CU4R9M 10413666 IC50 = 66 nM T85943 CHPR58 10416818 IC50 = 5300 nM T85943 CP6N2J 10423146 IC50 > 50000 nM T85943 C4CP7K 10423452 IC50 = 12900 nM T85943 C3MI7D 10430804 IC50 > 100000 nM T85943 CFLH53 10432113 IC50 = 19.95 nM T85943 CN5BF4 10434923 IC50 > 100000 nM T85943 C7QU9X 10437879 IC50 > 50000 nM T85943 CW75SO 10438950 IC50 = 0.3 nM T85943 CXA85V 10439212 IC50 = 7100 nM T85943 CZW1F0 10439643 IC50 = 2300 nM T85943 CEU25H 10445729 IC50 > 50000 nM T85943 CUX75O 10450005 IC50 > 50000 nM T85943 CT42KE 10450849 IC50 > 50000 nM T85943 CL7PF2 10451087 IC50 = 10 nM T85943 CSAZ29 10454329 IC50 = 38 nM T85943 C2Z8XR 10455073 IC50 = 20 nM T85943 C95LYF 10457505 IC50 > 30000 nM T85943 CY9DS7 10458235 IC50 = 433 nM T85943 CDQO71 10461517 IC50 = 3600 nM T85943 CW23SQ 10468973 IC50 > 50000 nM T85943 CH4CY9 10471016 IC50 = 19.95 nM T85943 C17OFQ 10476638 Ki = 3700 nM T85943 CR07PO 10477008 IC50 > 50000 nM T85943 CJ5M1D 10482445 IC50 = 20 nM T85943 COW2Q5 10483554 IC50 > 100000 nM T85943 C0EV8B 10494548 IC50 > 100000 nM T85943 C8DH5W 10499619 IC50 > 10000 nM T85943 C78FPR 10501266 IC50 = 2200 nM T85943 CSR8Y5 10527068 IC50 = 89000 nM T85943 CA0X6F 10531654 IC50 = 100 nM T85943 CHUY02 10555274 IC50 = 18400 nM T85943 C95ALZ 10555601 IC50 = 1600 nM T85943 CJW04C 10556625 IC50 = 6100 nM T85943 CW16DN 10568777 IC50 > 100000 nM T85943 CX67AG 10569366 IC50 > 100000 nM T85943 CP8J4O 10590515 IC50 > 100000 nM T85943 COB2X8 10602350 IC50 = 2200 nM T85943 CC8X4T 10603806 IC50 = 1400 nM T85943 C0LHE5 10615400 IC50 > 100000 nM T85943 CNE92Q 10616753 IC50 > 100000 nM T85943 C6VRE8 10626163 IC50 = 9100 nM T85943 CU8Q5N 10626988 IC50 = 17800 nM T85943 CUIN35 10629055 IC50 > 100000 nM T85943 CZ8UA9 10650891 IC50 > 100000 nM T85943 CNC85V 10651406 IC50 = 2700 nM T85943 CZ78VR 10660240 IC50 > 100000 nM T85943 CE6M3B 10674206 IC50 = 13000 nM T85943 CBX1F5 10674779 IC50 = 5000 nM T85943 CWVJ32 10677602 IC50 = 22800 nM T85943 CAVX96 10686149 IC50 > 100000 nM T85943 CK85TP 10692159 IC50 > 100000 nM T85943 CU8HZ7 10695922 IC50 = 30000 nM T85943 C18YJD 10698535 IC50 = 5700 nM T85943 CZP40T 10699325 IC50 = 3500 nM T85943 CU6G5Y 10708835 IC50 > 100000 nM T85943 C83QWV 10714343 IC50 = 8620 nM T85943 CCN2Q5 10721885 IC50 = 8600 nM T85943 CA4FT1 10722796 IC50 = 1000 nM T85943 CZVK65 10729749 IC50 > 100000 nM T85943 CJO8Q1 10738332 IC50 = 77 nM T85943 CL8VH3 10768554 IC50 > 100000 nM T85943 CQK0Z7 10769900 IC50 = 8100 nM T85943 C1OXH6 10803234 IC50 = 8000 nM T85943 COY52V 10812007 IC50 > 100000 nM T85943 C18MDA 10848423 IC50 > 100000 nM T85943 CI5FC1 10875157 IC50 = 7600 nM T85943 CJ4P5T 10905857 IC50 > 30000 nM T85943 CJ05CL 11048367 IC50 > 30000 nM T85943 CUT3V1 11125114 IC50 = 556 nM T85943 CH2KY3 11153440 Ki = 2400 nM T85943 CG9LZ6 11153921 Ki = 3600 nM T85943 CJ7U4I 11161778 IC50 < 50000 nM T85943 CN2JQ0 11169051 IC50 = 1400 nM T85943 CKZ31S 11178204 IC50 = 19 nM T85943 CD9E2W 11188787 IC50 = 2 nM T85943 C0Y8TX 11192751 IC50 = 35 nM T85943 CEUR60 11192985 IC50 = 77 nM T85943 C0L4GE 11199718 Ki = 1700 nM T85943 CB06ZF 11204217 IC50 = 240 nM T85943 C8G5WP 11210533 IC50 = 490 nM T85943 CEJ6F2 11214762 IC50 = 360 nM T85943 CF2GE5 11222252 Ki = 3000 nM T85943 C30NZT 11227609 IC50 = 25700 nM T85943 CH7D3X 11233762 IC50 = 3700 nM T85943 CVOW82 11238420 IC50 = 33900 nM T85943 C9RZV8 11245828 Ki = 630.96 nM T85943 C13MSX 11255450 Ki = 10000 nM T85943 CAHL14 11268810 Ki = 2900 nM T85943 CNBX16 11270660 IC50 = 20 nM T85943 CEP0G1 11273105 IC50 = 49 nM T85943 C8O2TU 11278922 Ki = 5011.87 nM T85943 C98TVJ 11279721 Ki = 10000 nM T85943 CJTP13 11280103 IC50 = 90000 nM T85943 CO2E3W 11280238 IC50 = 3000 nM T85943 CM9VK5 11281684 Ki = 7943.28 nM T85943 C30ALK 11291864 Ki = 1995.26 nM T85943 CBOP58 11293798 Ki > 10000 nM T85943 C9S8PK 11295293 IC50 = 1000 nM T85943 CANY24 11311217 IC50 > 100000 nM T85943 CRD9E5 11314043 IC50 = 9800 nM T85943 CMXI90 11324412 Ki = 2000 nM T85943 CIL0J6 11326339 Ki = 500 nM T85943 CD6X5Q 11329912 IC50 = 13 nM T85943 C04MZA 11331005 IC50 = 76300 nM T85943 CU5P8C 11331007 IC50 = 180 nM T85943 CKY3E2 11338122 IC50 > 100000 nM T85943 CUI2X1 11347617 Ki = 3162.28 nM T85943 C69ZAR 11360252 Ki = 2511.89 nM T85943 C26BZX 11362471 Ki > 10000 nM T85943 CGN8P2 11365768 IC50 = 70 nM T85943 CQ1Y5T 11370906 Ki = 1995.26 nM T85943 C3OCV2 11371778 IC50 = 4900 nM T85943 CQ40NG 11371816 Ki = 2400 nM T85943 C43NPS 11373886 IC50 > 10000 nM T85943 C25ZCN 11374110 IC50 > 50000 nM T85943 CUC0H2 11376301 IC50 > 100000 nM T85943 CT6Y9W 11376799 IC50 = 160 nM T85943 CZXI30 11384079 Ki = 7943.28 nM T85943 C6HBF0 11393275 Ki = 2400 nM T85943 CWXB93 11397177 Ki > 10000 nM T85943 C0LG2Y 11416582 Ki = 6309.57 nM T85943 C5O1RM 11421633 IC50 = 100 nM T85943 C0APW4 11422034 IC50 = 1100 nM T85943 CREQ51 11429654 IC50 > 50000 nM T85943 CY0A4E 11429729 IC50 > 50000 nM T85943 C3O0WI 11438191 IC50 = 90000 nM T85943 CWBJ70 11439347 IC50 = 11 nM T85943 C3EXM4 11440028 IC50 = 15700 nM T85943 CO4F0R 11443738 IC50 = 1700 nM T85943 CKM8E6 11444953 IC50 = 44 nM T85943 CWI62M 11454712 IC50 > 1000 nM T85943 CU50OG 11455909 IC50 = 160 nM T85943 COAZ38 11465148 IC50 = 9 nM T85943 C6L3AE 11473434 Ki = 2400 nM T85943 C7I6AG 11474111 IC50 = 78000 nM T85943 CS6GR3 11477850 IC50 = 8 nM T85943 CPC9S5 11489476 IC50 = 1900 nM T85943 C0H6QS 11495680 IC50 > 10000 nM T85943 C59LGV 11496101 IC50 = 118 nM T85943 CT9V3D 11496376 IC50 = 4000 nM T85943 CIF72P 11498974 IC50 > 700000 nM T85943 CBUK10 11501879 IC50 = 110 nM T85943 CIW9L5 11502867 IC50 > 10000 nM T85943 C52UMC 11507510 IC50 = 1500 nM T85943 CRU9D3 11508262 Ki = 2800 nM T85943 CEMK79 11513546 IC50 = 5600 nM T85943 CK2Q0X 11516978 IC50 > 10000 nM T85943 C8AY3B 11518031 IC50 < 25 nM T85943 CY2P5M 11520904 IC50 = 780 nM T85943 C3OPV8 11524973 IC50 = 15 nM T85943 CPE53F 11526238 IC50 > 10000 nM T85943 CHN68E 11530772 IC50 > 50000 nM T85943 CL7X4Q 11530963 IC50 = 20000 nM T85943 C5BM4T 11531799 IC50 > 10000 nM T85943 C53OSD 11532048 IC50 > 10000 nM T85943 CC4QM5 11532676 IC50 > 10000 nM T85943 C7KUJ3 11537047 IC50 = 269 nM T85943 CTG83F 11539329 Ki > 1900 nM T85943 CT64NL 11540547 IC50 = 0.75 nM T85943 CST9H8 11541124 IC50 = 31 nM T85943 CI23VD 11541324 IC50 = 14 nM T85943 CE9JR6 11542492 IC50 = 26000 nM T85943 CAT8P0 11545984 Ki = 3162.28 nM T85943 C01FVM 11546457 IC50 > 10000 nM T85943 CNX1C2 11549767 IC50 = 1400 nM T85943 C0E9IV 11554258 IC50 = 6 nM T85943 C9AK0U 11560211 IC50 > 50000 nM T85943 CACS26 11561968 Ki > 4000 nM T85943 CNBM81 11562171 IC50 > 10000 nM T85943 CJV20L 11569758 IC50 = 5.2 nM T85943 CPD3F8 11571561 IC50 = 75000 nM T85943 C9XI8Z 11574885 IC50 = 442 nM T85943 CMF8V4 11578809 IC50 = 93000 nM T85943 CPW27V 11581044 Ki = 1320 nM T85943 C8KUI7 11581459 IC50 > 50000 nM T85943 CG3N9Z 11581460 IC50 = 960 nM T85943 CO9KP5 11583459 IC50 > 10000 nM T85943 CAJQ78 11584678 IC50 = 3.6 nM T85943 C70NFR 11586052 IC50 = 10800 nM T85943 C3K8VD 11586070 IC50 > 400000 nM T85943 C9CS2E 11588163 IC50 = 40 nM T85943 C3VUO7 11588815 IC50 > 12500 nM T85943 CA2KX0 11590078 IC50 > 50000 nM T85943 CMIL86 11590363 Ki > 1900 nM T85943 CEAX60 11593162 IC50 = 760000 nM T85943 CKV24X 11593177 IC50 = 7300 nM T85943 CSYV06 11595313 IC50 > 50000 nM T85943 C6REV9 11595922 IC50 = 130 nM T85943 C0NV9Y 11596881 IC50 > 10000 nM T85943 C1TNR8 11602995 Ki = 10000 nM T85943 CYPD01 11603131 IC50 > 50000 nM T85943 C69FYK 11604142 Ki = 770 nM T85943 C43JZU 11604436 IC50 > 20000 nM T85943 CGU7N0 11604739 IC50 > 20000 nM T85943 COW68T 11605551 IC50 > 100000 nM T85943 CKW49P 11605989 IC50 = 10 nM T85943 C0FVM8 11610798 Ki = 1584.89 nM T85943 CJU5W6 11611103 Ki = 480 nM T85943 CV8L4F 11614881 IC50 = 54500 nM T85943 CQ89TH 11617657 Ki = 9600 nM T85943 C1BLZ5 11620055 IC50 > 10000 nM T85943 C5B3XJ 11620410 IC50 = 720 nM T85943 C4U7HM 11621097 IC50 = 53 nM T85943 C9ZD2E 11626406 IC50 = 914 nM T85943 C2QO0E 11626891 IC50 = 13 nM T85943 CSM62L 11626920 IC50 > 30000 nM T85943 CK34LS 11632737 IC50 > 10000 nM T85943 CBE73K 11634416 IC50 = 21 nM T85943 C9T6SC 11640926 Ki > 1900 nM T85943 CYBE19 11643683 IC50 > 700000 nM T85943 C8SIO0 11643703 IC50 = 134000 nM T85943 CW6D5K 11646082 IC50 = 180 nM T85943 CI4A8T 11650224 IC50 = 3.6 nM T85943 CQN26T 11660482 Ki = 2800 nM T85943 C1AUX0 11661290 IC50 = 396 nM T85943 C24GRQ 11661959 IC50 > 10000 nM T85943 CAJS96 11662893 IC50 > 20000 nM T85943 C9SL1J 11669430 Ki = 0.449 nM T85943 CKAH36 11669784 IC50 > 20000 nM T85943 CL8MO0 11672456 IC50 = 3400 nM T85943 CI72AM 11672471 IC50 > 400000 nM T85943 CX7H6I 11672472 IC50 = 1900 nM T85943 CM5D0R 11674900 Ki = 794.33 nM T85943 CU1FR7 11675061 IC50 > 50000 nM T85943 CCPZ18 11676103 IC50 = 140 nM T85943 COJ1F3 11680937 Ki = 10000 nM T85943 CS72ED 11682843 IC50 > 10000 nM T85943 CP3U0W 11684933 IC50 = 45 nM T85943 CSF35X 11685347 IC50 = 3.6 nM T85943 CSAL37 11686627 IC50 = 6000 nM T85943 CU0E8O 11690457 Ki > 4000 nM T85943 CO4PG2 11691040 IC50 = 10 nM T85943 CLC53E 11691173 IC50 > 10000 nM T85943 CLMS93 11693602 IC50 = 33600 nM T85943 CGVI01 11696703 Ki = 1584.89 nM T85943 C3MWR6 11696909 IC50 > 50000 nM T85943 C3JAX8 11699351 IC50 = 12 nM T85943 C9PZ3V 11702481 IC50 = 349 nM T85943 CB0AP2 11705863 Ki > 4000 nM T85943 CS16YM 11712202 IC50 = 10 nM T85943 CHL5W3 11712625 Ki = 1.3 nM T85943 C13YGW 11713440 IC50 = 25 nM T85943 CIDP74 11714929 IC50 = 1500 nM T85943 CHU25R 11715040 IC50 = 1000 nM T85943 CE49IU 11718919 Ki > 4000 nM T85943 C1FTX3 11719305 IC50 > 10000 nM T85943 CZY05V 11719421 IC50 = 6.4 nM T85943 C2Z8AE 11722068 IC50 > 700000 nM T85943 CMO03N 11722100 IC50 = 2000 nM T85943 CZ37XK 11722102 Ki = 210 nM T85943 CPIH89 11722723 IC50 = 800000 nM T85943 CFJ4I7 11723151 IC50 = 1600 nM T85943 C9HC4M 11726643 IC50 > 100000 nM T85943 C9P0VD 11729539 IC50 > 30000 nM T85943 CCX53Q 11729563 IC50 = 83000 nM T85943 C7C2FM 11737638 IC50 > 100000 nM T85943 CPY1Z2 11740563 IC50 < 1 nM T85943 COX34W 11741081 Ki = 600 nM T85943 CS9WP2 11752657 IC50 = 15 nM T85943 CN8S1E 11752715 IC50 = 440 nM T85943 CE0KI4 11753519 IC50 = 19700 nM T85943 CP7AH3 11755812 IC50 = 50000 nM T85943 CWL34S 11756855 IC50 = 2600 nM T85943 CCG4J6 11764871 IC50 = 18000 nM T85943 C3Q9WC 11764957 IC50 = 8600 nM T85943 CYBS49 11773690 Ki = 6309.57 nM T85943 C3J7MT 11777791 IC50 > 50000 nM T85943 CGYV23 11779501 IC50 > 50000 nM T85943 CL87KR 11785748 IC50 = 210 nM T85943 CV5EZ3 11798263 IC50 = 6500 nM T85943 CM10YB 11799388 IC50 = 11000 nM T85943 C9NH8P 11799946 IC50 = 12000 nM T85943 CJVR85 11802701 IC50 > 10000 nM T85943 CCI6R5 11842847 IC50 = 13 nM T85943 CMO6N4 11842849 IC50 = 98 nM T85943 C9HT7B 11842850 IC50 = 500 nM T85943 CP6KY2 11843009 IC50 = 1 nM T85943 C8FHK9 11843010 IC50 = 4 nM T85943 C7D6MQ 11843012 IC50 = 2 nM T85943 C4T2WC 11843013 IC50 = 2 nM T85943 CS36BH 11843159 IC50 = 1 nM T85943 C7DU6T 11843160 IC50 = 12 nM T85943 CH6W3V 11844349 IC50 = 10 nM T85943 CI15NA 11844350 IC50 = 3 nM T85943 CUL2C8 11844485 IC50 = 14 nM T85943 C96ORQ 11844486 IC50 = 2 nM T85943 C4SK3L 11844487 IC50 = 2 nM T85943 C6KF8Z 11844488 IC50 = 4 nM T85943 C9ECK3 11844489 IC50 = 1 nM T85943 C83YRX 11844616 IC50 = 5 nM T85943 CV24WL 11844764 IC50 = 4 nM T85943 CQF23E 11952856 IC50 = 11 nM T85943 CS81MP 11957378 IC50 = 68 nM T85943 CSC8A9 11973903 IC50 = 300 nM T85943 CK91AC 11973905 IC50 = 400 nM T85943 C8CJD5 11973906 IC50 = 100 nM T85943 CQ6J4I 11973907 IC50 = 230 nM T85943 CB60GC 11974016 IC50 = 750 nM T85943 CZG6O4 11974017 IC50 = 40 nM T85943 CUBL61 11974019 IC50 = 150 nM T85943 C15HWQ 11974020 IC50 = 6400 nM T85943 CYLH02 11974021 IC50 = 800 nM T85943 C2RSN3 11974115 IC50 = 1100 nM T85943 CY37WX 11974116 IC50 = 75 nM T85943 C0RB2T 11974118 IC50 = 500 nM T85943 CR3P7C 11974119 IC50 = 100 nM T85943 CXQ7Y1 11974120 IC50 = 4 nM T85943 C3Z1JF 11974212 IC50 = 7 nM T85943 C5OX6U 11974213 IC50 < 4 nM T85943 CF2P7Z 11974214 IC50 = 5 nM T85943 C0GZL5 11974215 IC50 = 200 nM T85943 CYM4Q5 11974217 IC50 = 3000 nM T85943 C9XOP3 11974219 IC50 = 3700 nM T85943 COFI19 11974316 IC50 = 764 nM T85943 C1TX8I 11974329 IC50 = 600 nM T85943 CS0ZM6 11974330 IC50 = 110 nM T85943 CIB76J 11974331 IC50 = 65 nM T85943 CHUA95 11974417 IC50 = 3.9 nM T85943 CF78KB 12241337 IC50 = 4000000 nM T85943 C7EV4K 12241338 IC50 = 2000000 nM T85943 C9MHX7 12484326 IC50 > 50000 nM T85943 CSGC17 12499981 IC50 = 4000000 nM T85943 C5CPV2 12516472 IC50 > 20 ug.mL-1 T85943 C1W9RA 12741204 IC50 = 4000000 nM T85943 COIJ48 12968819 IC50 = 459000 nM T85943 C4AIU2 12968822 IC50 = 205000 nM T85943 CWUK08 13492269 IC50 > 100000 nM T85943 C2QEX8 13492281 IC50 > 100000 nM T85943 C1D0WF 14362924 Ki = 605 nM T85943 C2N3WV 14638906 Ki = 500 nM T85943 CUMI23 14943555 IC50 = 16300 nM T85943 CRZG26 14943556 IC50 = 7900 nM T85943 C5M6ZT 14943557 IC50 = 5500 nM T85943 CW48TD 15159374 IC50 = 5290 nM T85943 C3SYC4 15159375 IC50 = 294 nM T85943 C7V5WC 15159376 IC50 = 387 nM T85943 CQ49GK 15159377 IC50 = 3500 nM T85943 C3FH4K 15159378 IC50 = 852 nM T85943 C0KQD6 15159379 IC50 = 820 nM T85943 C95SKG 15159380 IC50 = 477 nM T85943 CJKX79 15159381 IC50 = 436 nM T85943 C2DKN0 15159382 IC50 > 27000 nM T85943 CK8XF4 15209376 IC50 > 100000 nM T85943 CPK05U 15249955 IC50 > 100000 nM T85943 CDGF78 15282555 IC50 = 1900 nM T85943 C3YRU7 15295578 IC50 > 50000 nM T85943 CU6VD7 15366660 IC50 > 10000 nM T85943 CIL1R3 15411595 IC50 = 1200 nM T85943 CI4U8X 15549009 IC50 = 32000 nM T85943 C7N6CQ 15604547 IC50 = 480 nM T85943 CP8OW6 15858662 IC50 = 50.12 nM T85943 CUI6E5 15858664 IC50 = 1 nM T85943 C6PZU3 15858665 IC50 = 19.95 nM T85943 CEMH32 15858666 IC50 = 6 nM T85943 CK5QI3 15858667 IC50 = 53 nM T85943 CXZ0O1 15858769 IC50 = 800 nM T85943 C4I3PF 15858771 IC50 = 3400 nM T85943 C4VI8S 15927977 IC50 = 3500000 nM T85943 C0M7TW 15948947 IC50 = 107 nM T85943 C1VNB4 15948949 IC50 = 39 nM T85943 CH8ZG5 15949048 IC50 = 57 nM T85943 CK2Z6Y 15949521 IC50 = 1539 nM T85943 CBZF29 15949522 IC50 = 1650 nM T85943 C34MCY 15949523 IC50 = 47 nM T85943 CS3P9G 15949524 IC50 = 32 nM T85943 C1KPH2 15949525 IC50 = 16507 nM T85943 C7LB4I 15949613 IC50 > 10000 nM T85943 C5JG9R 15949617 IC50 = 4 nM T85943 C8FT6U 15949618 IC50 = 959 nM T85943 C30PVQ 15949619 IC50 = 7359 nM T85943 C3PNO2 15949620 IC50 = 177 nM T85943 C4I5RS 15949621 IC50 > 2500 nM T85943 CVJ9A0 15949712 IC50 = 5 nM T85943 CEI2K8 15949887 IC50 = 147 nM T85943 CAIN63 15949888 IC50 > 2500 nM T85943 C2VDI1 15949889 IC50 = 1698 nM T85943 COC02T 15949890 IC50 = 1378 nM T85943 CFQ6X3 15949974 IC50 = 918 nM T85943 CMKZ23 15949975 IC50 = 398 nM T85943 CWM5L4 15949976 IC50 = 601 nM T85943 CO7NG2 15950141 IC50 = 97 nM T85943 COIG45 15950224 IC50 = 450 nM T85943 C9V0TO 15950311 IC50 > 10000 nM T85943 C9TS5M 15950818 IC50 = 52000 nM T85943 CFPW41 16007116 Ki > 1900 nM T85943 CZTN89 16040366 IC50 = 9 nM T85943 CQR5O7 16042971 IC50 > 10000 nM T85943 CN36QI 16043219 IC50 = 3 nM T85943 C9JK2M 16059071 IC50 = 1500 nM T85943 CW6UJ9 16059338 IC50 = 1000 nM T85943 CH7MS6 16059729 IC50 = 5900 nM T85943 CFKE48 16064750 IC50 > 6000 nM T85943 CYWC40 16071691 IC50 > 10000 nM T85943 CKX2L7 16085320 IC50 = 3000 nM T85943 CKR57M 16086104 IC50 = 17 nM T85943 C16NRY 16086114 IC50 = 2 nM T85943 C3TQ4R 16099168 IC50 = 2.7 nM T85943 CBLR89 16099169 IC50 = 7.5 nM T85943 CSX2W1 16099173 IC50 = 11 nM T85943 C8HI5N 16099174 IC50 = 2800 nM T85943 CCWL52 16099179 IC50 = 13 nM T85943 CQG45C 16109001 IC50 = 5750 nM T85943 CGC34R 16118737 IC50 = 3 nM T85943 C6H4ZW 16126744 IC50 = 950 nM T85943 CP3HS4 16220354 IC50 = 30400 nM T85943 CJ5KU9 16659012 IC50 = 830 nM T85943 C6TQ2O 16664354 Ki = 7.22 nM T85943 CU56EW 16664858 IC50 > 10000 nM T85943 C2IF3P 16678352 IC50 = 5300 nM T85943 C3IO1C 16679060 IC50 = 770 nM T85943 CN1YG9 16720859 IC50 > 100000 nM T85943 C2AI5C 16741056 IC50 > 100000 nM T85943 CU7ME4 16743447 IC50 = 175 nM T85943 C5LV3Z 16743632 IC50 = 408 nM T85943 CZS76J 16744317 IC50 = 2990 nM T85943 CDZ31W 16747696 IC50 > 50000 nM T85943 CL9BQ6 17748275 IC50 = 2195 nM T85943 CVS0T5 17754396 IC50 > 10000 nM T85943 CAV9R6 17757434 IC50 = 38000 nM T85943 C8AH1I 17758019 IC50 = 40800 nM T85943 C1GKL6 17758020 IC50 > 40000 nM T85943 CIE58R 17758239 IC50 > 40000 nM T85943 CO6LR5 17758240 IC50 = 20000 nM T85943 CWH37T 17758574 IC50 > 40000 nM T85943 C9VLS2 17759429 IC50 = 5400 nM T85943 C57NRL 17759787 IC50 > 40000 nM T85943 CQ35AK 17953498 IC50 = 100 nM T85943 CJA0D6 18451024 IC50 = 14400 nM T85943 C6FQB7 18451036 IC50 = 9050 nM T85943 CG21ZB 18455722 IC50 > 50000 nM T85943 C02LRI 18455757 IC50 = 2200 nM T85943 CDT3U6 18455762 IC50 = 12000 nM T85943 CQN96H 18731516 IC50 = 1370700 nM T85943 C1C0EJ 18792861 IC50 = 1 nM T85943 C6HK0S 18792868 IC50 = 3 nM T85943 C90EQY 18792940 IC50 = 37 nM T85943 C9PS7R 18792941 IC50 = 25.12 nM T85943 CIH2K0 18792942 IC50 = 4 nM T85943 CY5N7Z 18792945 IC50 = 300 nM T85943 CILQ48 18792962 IC50 = 230 nM T85943 CU5CK6 19597400 IC50 > 1000 nM T85943 CZQ92B 19597433 IC50 = 48 nM T85943 CIBE65 19597460 IC50 = 1470 nM T85943 CP01WN 19597468 IC50 = 40 nM T85943 C0WEX3 19966997 IC50 > 100000 nM T85943 CJC5F3 20741385 Ki = 2984 nM T85943 CV7C2K 20817018 IC50 = 97 nM T85943 CQ5X7V 20817081 IC50 = 56 nM T85943 CJN28H 21014352 IC50 = 16000 nM T85943 CV6AB7 21036218 IC50 = 150000 nM T85943 CA61QF 21083895 IC50 < 50000 nM T85943 CUL91S 21879790 IC50 > 10000000 nM T85943 CQY89R 21980377 IC50 = 46000 nM T85943 CTAO10 21980612 IC50 = 17000 nM T85943 CT3QM7 21980728 IC50 = 27000 nM T85943 C8IF5U 21991073 Ki = 2180 nM T85943 CQ2XW6 22346679 IC50 = 17150 nM T85943 CXEW46 22500191 IC50 = 3300 nM T85943 CLOR96 22736225 IC50 = 390 nM T85943 CT39NL 22736235 IC50 = 88 nM T85943 CAU62I 22736238 IC50 = 32340 nM T85943 CV1OI5 22736332 IC50 = 320 nM T85943 C5ONK2 22736361 IC50 = 1120 nM T85943 C0HRM6 22911602 IC50 = 11000 nM T85943 C8UPY9 23437830 IC50 = 36 nM T85943 CDHQ58 23437865 IC50 = 950 nM T85943 CF65HC 23437877 IC50 = 24 nM T85943 C1QKM4 23438122 IC50 = 4 nM T85943 CUS3A4 23438137 IC50 = 170 nM T85943 CH5UC4 23438375 IC50 = 26 nM T85943 CHF1K3 23518506 IC50 = 300 nM T85943 CG12OL 23518511 IC50 = 70 nM T85943 CE7K3W 23532567 IC50 > 10000 nM T85943 COW62H 23646038 IC50 = 250 nM T85943 COB95G 23646040 IC50 = 15 nM T85943 CQHK69 23646624 IC50 = 710 nM T85943 C2PKU9 23646845 IC50 = 300000 nM T85943 C2JTA3 23647573 IC50 > 50000 nM T85943 C17HUI 23647581 IC50 = 18000 nM T85943 C2C3EM 23649898 IC50 = 300000 nM T85943 CML17W 23655479 Ki = 4000 nM T85943 C7MT4E 23655480 Ki = 15000 nM T85943 CWV5K4 23655678 Ki = 2800 nM T85943 CI9PE2 23655679 Ki = 3100 nM T85943 CT0SZ7 23655680 Ki = 21000 nM T85943 CVW9M8 23655681 Ki = 3000 nM T85943 C1MDZ7 23655682 Ki = 600 nM T85943 C10KDP 23655683 Ki = 1800 nM T85943 CF3A7U 23655878 Ki = 500 nM T85943 C5TV4F 23655879 Ki = 4100 nM T85943 C6JTW3 23656073 Ki = 13000 nM T85943 CGIH32 23656074 Ki = 6000 nM T85943 C7IU1G 23656075 Ki = 25000 nM T85943 C3GWO1 23656076 Ki = 4000 nM T85943 C4F1VE 23656077 Ki = 7500 nM T85943 CI3T7F 23656078 Ki = 24000 nM T85943 C7TG0V 23656262 Ki = 5200 nM T85943 CE5XF1 23656263 Ki = 4600 nM T85943 C64ESF 23656264 Ki = 35000 nM T85943 CGC07X 23656265 Ki = 1400 nM T85943 C8B7PK 23656266 Ki = 1200 nM T85943 CN17BU 23656267 Ki = 1200 nM T85943 C4JE1L 23657441 IC50 = 3.5 nM T85943 CI6C1R 23658582 IC50 = 117 nM T85943 C6O8QY 23661616 IC50 = 1.5 nM T85943 C2S5ZM 23661662 Ki = 27 nM T85943 CUGY24 24202429 IC50 = 800 nM T85943 CY75PZ 24757723 IC50 > 10000 nM T85943 C7YG1N 24759534 IC50 = 37 nM T85943 CAJ4T2 24762205 IC50 = 662 nM T85943 CQNP54 24764449 IC50 = 1000 nM T85943 CCPS81 24764502 IC50 > 35000 nM T85943 C2UOE0 24766030 IC50 = 330 nM T85943 CJUK39 24770517 IC50 > 10000 nM T85943 C0EKO5 24772654 IC50 = 58 nM T85943 CB9N8E 24802574 Ki = 800 nM T85943 CQK54U 24807247 Ki = 151 nM T85943 C5CXU0 24807250 Ki = 1500 nM T85943 C1B8AS 24807618 Ki = 500 nM T85943 CS6DA5 24807619 Ki = 80 nM T85943 C0JUN4 24812717 IC50 = 400 nM T85943 CP6N9M 24812718 IC50 = 5000 nM T85943 CW0G8H 24812719 IC50 = 860 nM T85943 CCP2M3 24822704 IC50 > 50000 nM T85943 CCON58 24822755 IC50 > 50000 nM T85943 C7GWU6 24822756 IC50 = 7400 nM T85943 C48RDH 24822757 IC50 = 3600 nM T85943 CV0O7Y 24822918 IC50 = 778 nM T85943 C2MUA7 24823072 IC50 = 340 nM T85943 CX94DT 24823073 Ki = 35 nM T85943 C3A2BF 24823416 IC50 = 8300 nM T85943 CG0K1Z 24824046 IC50 = 240 nM T85943 CS82HN 24856408 IC50 = 1000 nM T85943 CZ5Y4H 24856498 IC50 = 462 nM T85943 CC10FW 24857629 IC50 > 1000 nM T85943 C7BU8A 24864305 IC50 > 10000 nM T85943 CJ0XU5 24864851 IC50 > 10000 nM T85943 C0Z8VJ 24866469 IC50 = 580 nM T85943 CV21ZF 24879059 IC50 = 4500 nM T85943 CG13IK 24879061 IC50 = 1700 nM T85943 CJ6TN2 24879098 IC50 = 8400 nM T85943 CE3IW4 24879184 IC50 = 260 nM T85943 C7V8BA 24879242 IC50 = 390 nM T85943 CT76XV 24879243 IC50 = 43 nM T85943 CGD8J5 24879244 IC50 = 170 nM T85943 C1XWO7 24879245 IC50 = 77 nM T85943 CA21RX 24879305 IC50 = 800 nM T85943 COF05N 24879306 IC50 = 990 nM T85943 C6NIQ2 24879307 IC50 = 36 nM T85943 C45HIT 24879308 IC50 = 750 nM T85943 CM6G7A 24879309 IC50 = 150 nM T85943 C0KW5Y 24879310 IC50 = 270 nM T85943 C7M9FB 24879311 IC50 = 25000 nM T85943 C0ZJX6 24879366 IC50 = 390 nM T85943 C5NA4Z 24879367 IC50 = 1400 nM T85943 CDJE41 24879368 IC50 > 5000 nM T85943 C9B2TF 24880043 IC50 = 1400 nM T85943 CA8M5O 24880570 IC50 > 10000 nM T85943 CFK2B9 24882503 IC50 = 66 nM T85943 C43HWQ 24883287 IC50 = 800 nM T85943 C8DA5Q 24883334 IC50 < 100 nM T85943 C13QYB 24884503 IC50 > 2000 nM T85943 CQ3S5Y 24884916 IC50 = 31000 nM T85943 CWAL41 24885316 IC50 = 5600 nM T85943 C0P6AU 24894017 IC50 < 1 nM T85943 C4V9GH 24894117 IC50 = 14000 nM T85943 CHVU39 24894885 IC50 = 39000 nM T85943 CZ6KD4 24894886 IC50 = 4500 nM T85943 C57BHF 24894888 IC50 = 40000 nM T85943 CB5TP8 24894992 IC50 = 4400 nM T85943 C32SUJ 24894993 IC50 = 9100 nM T85943 CP7QT2 24894995 IC50 = 41000 nM T85943 C41SIT 24894996 IC50 = 29000 nM T85943 CFW40U 24894997 IC50 = 49000 nM T85943 CY8L7E 24896769 IC50 > 10000 nM T85943 CN13JF 24899915 IC50 = 5.6 ug.mL-1 T85943 CBWR97 24899916 IC50 = 1.4 ug.mL-1 T85943 C9F2JD 24899917 IC50 > 10 ug.mL-1 T85943 C64MTI 24900160 IC50 = 4.7 ug.mL-1 T85943 CO2I6Q 24900161 IC50 = 4.6 ug.mL-1 T85943 CB79YC 24905143 IC50 = 15 nM T85943 C2DC9J 24905144 IC50 = 1100 nM T85943 CN6V8Z 24905145 IC50 = 10 nM T85943 CSB7P5 24905148 IC50 = 11000 nM T85943 CGSF21 24905149 IC50 = 17000 nM T85943 CVDG02 24905150 IC50 < 1 nM T85943 CWH6C5 24905152 IC50 = 240 nM T85943 C0HE2Q 24905153 IC50 = 170 nM T85943 C7QSC9 24905154 IC50 = 3200 nM T85943 CO9D0K 24905155 IC50 = 2100 nM T85943 C5W9UR 24905157 IC50 = 1500 nM T85943 CC1DA3 24905158 IC50 = 5200 nM T85943 COW79F 24905159 IC50 = 7200 nM T85943 CFPA53 24905160 IC50 = 5900 nM T85943 C2O0JX 24905161 IC50 = 2300 nM T85943 CA72BE 24905162 IC50 = 5000 nM T85943 CQN6X9 24905163 IC50 = 12000 nM T85943 CD4O1F 24905165 IC50 = 3000 nM T85943 CKL48T 24905166 IC50 = 890 nM T85943 C76VYL 24905167 IC50 = 3000 nM T85943 C7K5PU 24905168 IC50 = 380 nM T85943 CZ57ID 24905169 IC50 = 160 nM T85943 C2DHX9 24905170 IC50 = 8700 nM T85943 CSB96E 24905171 IC50 = 50000 nM T85943 CWZ0R2 24905172 IC50 = 930 nM T85943 CY3B6M 24905175 IC50 = 98 nM T85943 CW7UA3 24905176 IC50 = 476 nM T85943 CW1V0H 24905177 IC50 = 76 nM T85943 CO6Y0L 24905178 IC50 = 499 nM T85943 C60NQW 24905179 IC50 = 1430 nM T85943 C4MO8B 24905180 IC50 = 25 nM T85943 COJI47 24905181 IC50 = 10 nM T85943 CS0B2C 24905182 IC50 = 5 nM T85943 C1H4BT 24905183 IC50 = 2.2 nM T85943 C4WHK9 24905184 IC50 = 286 nM T85943 C7Q4MZ 24905185 IC50 = 46 nM T85943 CS4IP1 24905186 IC50 = 31 nM T85943 C69QWO 24905187 IC50 = 194 nM T85943 C85ANB 24905188 IC50 = 39 nM T85943 CNHD75 24905189 IC50 = 180 nM T85943 C9JUO2 24905190 IC50 = 37 nM T85943 CPR03K 24905191 IC50 = 57 nM T85943 CTAG19 24905193 IC50 = 8 nM T85943 C7VJM5 24905194 IC50 = 1030 nM T85943 CEP1L3 24905195 IC50 = 238 nM T85943 CP68ZD 24905196 IC50 = 140 nM T85943 C8Z0RJ 24905197 IC50 = 135 nM T85943 CN9RT0 24905198 IC50 = 341 nM T85943 CHI78P 24905200 Ki = 200 nM T85943 CO6PE8 24905201 IC50 = 42 nM T85943 CZ63HS 24905202 IC50 = 20 nM T85943 C2X0FC 24905203 IC50 = 69 nM T85943 C0WCE3 24905204 IC50 = 12000 nM T85943 CNK50B 24905205 IC50 = 810 nM T85943 C12DPB 24905206 IC50 = 42 nM T85943 C8N0RH 24905207 IC50 = 2400 nM T85943 CYA5G2 24905208 IC50 = 100000 nM T85943 CDV2B4 24905209 IC50 = 250 nM T85943 CEFK68 24905210 IC50 = 440 nM T85943 CUFP12 24905211 IC50 = 716 nM T85943 C0JG8L 24905212 IC50 = 17 nM T85943 CQ13ZI 24905215 IC50 = 800 nM T85943 C6VI8F 24905216 IC50 = 2700 nM T85943 CXNH25 24905217 IC50 = 11000 nM T85943 C2PN9S 24905218 IC50 = 1000 nM T85943 C9O2AL 24905219 IC50 = 550 nM T85943 CIT7U8 24905220 IC50 = 2100 nM T85943 CMD26S 24905221 IC50 = 157 nM T85943 C4R8WC 24905222 IC50 = 211 nM T85943 C47SHA 24905223 IC50 = 73 nM T85943 C1DY2R 24905224 IC50 = 49 nM T85943 CS0XF9 24905225 IC50 = 30000 nM T85943 CG5VX2 24905226 IC50 = 7200 nM T85943 C57QEO 24905227 IC50 = 100000 nM T85943 C7CG5E 24905228 IC50 = 800 nM T85943 CHP5D1 24905229 IC50 = 1600 nM T85943 CXP09S 24905230 IC50 = 525 nM T85943 CY7XG1 24905231 IC50 = 12000 nM T85943 C7JFQ2 24905232 IC50 = 7600 nM T85943 C2JM1P 24905233 IC50 = 2700 nM T85943 CC3BF0 24905234 IC50 = 15000 nM T85943 CE57FI 24905235 IC50 = 764 nM T85943 CUP20O 24905236 IC50 = 1500 nM T85943 CLC6Q2 24905237 IC50 = 4400 nM T85943 C9M1GI 24905238 IC50 = 490 nM T85943 CVD72F 24905239 IC50 = 58 nM T85943 CK38IZ 24905240 IC50 = 408 nM T85943 CO2V5E 24905241 IC50 = 3500 nM T85943 CZBA19 24905244 IC50 = 103 nM T85943 CQ8OI1 24905246 IC50 = 23000 nM T85943 CIF2J5 24905251 IC50 = 23 nM T85943 CPTE58 24905252 IC50 = 40 nM T85943 C6XHJ7 24905272 Ki = 65 nM T85943 CP50RD 24905280 IC50 = 6.9 nM T85943 CG13ZM 24905281 IC50 = 11 nM T85943 CF0S6X 24905282 IC50 = 361 nM T85943 C5HBL0 24905284 IC50 = 33000 nM T85943 C2Z5DN 24905285 IC50 = 164 nM T85943 CL6GH8 24905286 IC50 = 489 nM T85943 CKYO98 24905287 IC50 = 4.3 nM T85943 CRNQ65 24905288 IC50 = 17 nM T85943 COD7I5 24905289 IC50 = 16 nM T85943 C4LP7E 24905290 IC50 = 96 nM T85943 CE9JC2 24905291 IC50 = 510 nM T85943 C2GI1R 24905292 IC50 = 100000 nM T85943 CHW8C4 24905293 IC50 = 67 nM T85943 CQF0H1 24905294 IC50 = 6.3 nM T85943 CNO7X0 24905295 IC50 = 4 nM T85943 C5WRG7 24905296 IC50 = 142 nM T85943 CQ1S0U 24905297 IC50 = 15200 nM T85943 C4UES7 24905298 IC50 = 175 nM T85943 CMS69P 24905299 IC50 = 132 nM T85943 CC0U5M 24905300 IC50 = 0.12 nM T85943 CW7X6S 24905301 IC50 = 747 nM T85943 C97IQV 24905302 IC50 = 0.55 nM T85943 CSJ47V 24905303 IC50 = 202 nM T85943 CPN74C 24905304 IC50 = 96 nM T85943 C5CS3N 24905305 IC50 = 25 nM T85943 CK4XE9 24905307 IC50 = 82 nM T85943 CTU6Z3 24905308 IC50 = 42 nM T85943 C9SQX1 24905309 IC50 = 15 nM T85943 CM75JP 24905310 IC50 = 46 nM T85943 C9Q2BJ 24905311 IC50 = 131 nM T85943 C9VUA1 24905312 IC50 = 30 nM T85943 CU3RS1 24905313 IC50 = 241 nM T85943 CYG3H2 24905314 IC50 = 17 nM T85943 CV5Q7O 24905315 IC50 = 1 nM T85943 C8SA3O 24905316 IC50 = 4 nM T85943 CI5MN3 24905317 IC50 = 2 nM T85943 CJ1P7K 24905318 IC50 = 7 nM T85943 C1T6YQ 24905319 IC50 = 14 nM T85943 CAU86X 24905320 IC50 = 31 nM T85943 C54ISY 24905321 IC50 = 101 nM T85943 C2GE5I 24905322 IC50 = 73 nM T85943 C8D6YK 24905323 IC50 = 405 nM T85943 C5NZH9 24905324 IC50 = 284 nM T85943 C9D6JR 24905325 IC50 = 24 nM T85943 CLZT41 24905326 IC50 = 11 nM T85943 CW8FD3 24905327 IC50 = 14 nM T85943 CHB7A2 24905328 IC50 = 90 nM T85943 CA8EI3 24905329 IC50 = 18 nM T85943 CCQ0O7 24905330 IC50 = 293 nM T85943 CJ81AS 24905331 IC50 = 61 nM T85943 C8PW4H 24905332 IC50 = 9.5 nM T85943 C2Y5TF 24905333 IC50 = 11 nM T85943 CH9FL5 24905334 IC50 = 3200 nM T85943 C1S0PC 24905335 IC50 = 3900 nM T85943 C8N9MV 24905336 IC50 = 72 nM T85943 C9E8BJ 24905338 IC50 = 11000 nM T85943 CX85AC 24905341 IC50 = 12000 nM T85943 CKZ80E 24905342 IC50 = 33 nM T85943 CO8SH1 24905343 IC50 = 530 nM T85943 C7IZL6 24905344 IC50 = 530 nM T85943 C5ZM4T 24936119 IC50 = 3 nM T85943 C5FD1A 24937369 IC50 = 1500 nM T85943 C15BZP 24949852 IC50 = 360 nM T85943 CZHE50 24949856 IC50 = 1600 nM T85943 C4V9GI 24960018 IC50 = 13200 nM T85943 CD5HQ0 24969301 IC50 > 10000 nM T85943 CBK82P 25011729 IC50 < 100 nM T85943 CZ7L3T 25022605 IC50 = 15.4 nM T85943 CX1HL8 25032704 Ki > 1940 nM T85943 C2ICS7 25065806 IC50 = 8.31 nM T85943 CQ67BO 25113172 Ki > 3330 nM T85943 CTV54O 25123227 IC50 > 10000 nM T85943 CIO41X 25169119 IC50 = 15 nM T85943 CAX51Q 25169120 IC50 = 50.6 nM T85943 CLCY94 25169121 IC50 = 267 nM T85943 CID5O7 25169255 Ki = 862 nM T85943 CN2B0H 25169256 Ki = 422 nM T85943 CTO24B 25174101 IC50 = 64100 nM T85943 CIG4H0 25178539 IC50 = 3800 nM T85943 CQ1E0N 25185128 Ki = 300 nM T85943 CP3EN4 25185129 Ki = 3250 nM T85943 CYN31L 25185130 Ki = 210 nM T85943 C40LQJ 25185131 Ki = 1320 nM T85943 C2PR9C 25185132 Ki = 1530 nM T85943 CF8GX1 25185133 Ki = 1620 nM T85943 CE4LB1 25185134 Ki = 3210 nM T85943 CUVP43 25185398 Ki = 3600 nM T85943 CH8J4V 25185399 Ki = 2560 nM T85943 COL73S 25185400 Ki = 510 nM T85943 CP6G0U 25185403 Ki = 810 nM T85943 C3FU2E 25185404 Ki = 1630 nM T85943 CZ80GV 25185687 Ki = 2570 nM T85943 CIU1P5 25185688 Ki = 220 nM T85943 CXQ10W 25185691 Ki = 4100 nM T85943 CZ60BO 25185692 Ki = 4220 nM T85943 CXMN65 25185693 Ki = 5280 nM T85943 C4L2VA 25185968 Ki = 5370 nM T85943 C1LIZ0 25185969 Ki = 2550 nM T85943 C81UNB 25185970 Ki = 5660 nM T85943 CX2IE4 25185971 Ki = 320 nM T85943 C94EPM 25185972 Ki = 2800 nM T85943 CH3X8S 25185973 Ki = 3630 nM T85943 CZG39U 25189269 Ki = 10200 nM T85943 CPZ70U 25189270 Ki = 2610 nM T85943 CF6GK9 25189271 Ki = 5020 nM T85943 C4QG2L 25189272 Ki = 3320 nM T85943 C7FMJ5 25189273 Ki = 310 nM T85943 CX3F4U 25195515 Ki = 700 nM T85943 CLFM35 25206064 IC50 > 50000 nM T85943 C6FGQ1 25206346 IC50 = 130 nM T85943 C41MJN 25210518 IC50 = 32100 nM T85943 CRO09K 25211064 IC50 = 55 nM T85943 C6L9FV 25211674 IC50 = 4 nM T85943 C3F7QN 25211675 IC50 = 5.56 nM T85943 C43UPC 25211772 IC50 = 0.89 nM T85943 C2TXC6 25218656 IC50 = 930 nM T85943 CK7ZR2 25242643 IC50 = 2900 nM T85943 CN5E0F 25263283 IC50 < 50000 nM T85943 CDWG95 25268881 IC50 = 82300 nM T85943 CC71QJ 27666048 IC50 > 100000 nM T85943 CHO43Y 28491869 IC50 = 1860 nM T85943 CIW8V3 40833444 Ki = 247 nM T85943 CVM13K 42596931 IC50 = 642 nM T85943 CS1AT2 42603881 IC50 = 75000 nM T85943 CZ2VH7 42604008 IC50 = 82000 nM T85943 C8B6TY 42628503 EC50 < 500 nM T85943 CI9DK5 42628614 IC50 = 500 nM T85943 CU9E4P 42629114 IC50 > 10000 nM T85943 CR5XJ4 42630202 IC50 = 89 nM T85943 CAR7C5 42631795 IC50 = 4200 nM T85943 CUY2S7 42631796 IC50 = 7400 nM T85943 CRD16V 42631905 IC50 = 3500 nM T85943 C7X9HZ 42632254 IC50 = 6500 nM T85943 C5Y1TL 42632378 IC50 = 5900 nM T85943 CS3T8Q 42632379 IC50 = 3300 nM T85943 CS5B4U 42632380 IC50 = 4900 nM T85943 C4TG6I 42632381 IC50 = 9900 nM T85943 CJ5U1X 42639664 IC50 = 1.7 ug.mL-1 T85943 CKG80R 42805643 Ki = 263 nM T85943 C48USC 44143344 IC50 = 40000 nM T85943 C8YN5P 44143370 IC50 = 53000 nM T85943 C9CWO1 44143371 IC50 = 72000 nM T85943 C26XFL 44143372 IC50 = 35000 nM T85943 C5SEQ2 44143373 IC50 = 110000 nM T85943 CTN41Y 44156909 IC50 > 10000 nM T85943 CN0X1C 44156917 IC50 > 10000 nM T85943 CLW80F 44160269 IC50 = 600 nM T85943 CBK37X 44195626 IC50 > 150000 nM T85943 C0FG6B 44198001 IC50 = 272100 nM T85943 C8KNA3 44219632 Ki > 4000 nM T85943 C0VIX4 44219633 Ki > 4000 nM T85943 CK73NR 44219749 IC50 > 50000 nM T85943 C1OJ5W 44221514 IC50 = 91000 nM T85943 C48QGV 44221515 IC50 = 4700 nM T85943 CWB74L 44221727 IC50 = 159000 nM T85943 CK5G4H 44221730 IC50 = 86000 nM T85943 C4H6WC 44221731 IC50 = 46000 nM T85943 CP3Z1S 44221732 IC50 = 46000 nM T85943 C2K5IO 44221929 IC50 = 84 nM T85943 C9LU0Y 44221931 IC50 = 45000 nM T85943 CB2A0O 44222109 IC50 = 201000 nM T85943 CXKZ46 44222110 IC50 = 9300 nM T85943 C4YS1K 44222111 IC50 = 26000 nM T85943 C54QWZ 44222112 IC50 = 3800 nM T85943 CV8P4L 44222285 IC50 = 11000 nM T85943 C7NK8F 44222286 IC50 = 4800 nM T85943 C42AML 44222458 IC50 = 310000 nM T85943 CK3S2I 44222459 IC50 = 6600 nM T85943 CJ43YR 44222636 IC50 = 517000 nM T85943 C65TLI 44222639 IC50 = 8000 nM T85943 CY5IU1 44222822 IC50 = 33000 nM T85943 C2MJI4 44222823 IC50 = 41000 nM T85943 C6MPO3 44222824 IC50 = 307 nM T85943 CEL61X 44229839 IC50 = 8400 nM T85943 CVH36D 44264208 IC50 = 105000 nM T85943 CTS57R 44268558 IC50 = 3900 nM T85943 CMN0Y1 44268559 IC50 = 20000 nM T85943 CZVK01 44268567 IC50 = 4600 nM T85943 COLK85 44268574 IC50 ~ 30000 nM T85943 C18AGO 44268577 IC50 = 6400 nM T85943 CR0Y8A 44268578 IC50 = 14000 nM T85943 CW19KH 44268584 IC50 ~ 46000 nM T85943 C9NA3E 44268603 IC50 = 12000 nM T85943 COJ62A 44268616 IC50 = 4300 nM T85943 CWPM51 44268618 IC50 = 4800 nM T85943 C1YA3K 44268619 IC50 = 10000 nM T85943 C04KJI 44268621 IC50 = 15000 nM T85943 CN47GT 44268631 IC50 = 10000 nM T85943 CDNP40 44268635 IC50 = 240 nM T85943 C85VMZ 44268654 IC50 = 3200 nM T85943 CABE60 44268655 IC50 = 2300 nM T85943 CC7YP6 44272770 IC50 = 3300 nM T85943 C8O4CU 44273012 IC50 = 13400 nM T85943 CGQ01B 44273030 IC50 = 21300 nM T85943 CVCB76 44273031 IC50 = 4000 nM T85943 CR2BZ3 44273189 IC50 = 30000 nM T85943 CEXF97 44273226 IC50 = 30000 nM T85943 CLEK41 44273227 IC50 = 40000 nM T85943 CQI7C8 44273228 IC50 = 30000 nM T85943 C9YAX6 44273229 IC50 = 28000 nM T85943 C3EFQ0 44273554 IC50 > 100000 nM T85943 CMRX16 44273620 IC50 > 100000 nM T85943 C9JB4G 44274666 IC50 = 2100000 nM T85943 CQA2U7 44274758 IC50 = 7800 nM T85943 C6JGV7 44274770 IC50 = 4500 nM T85943 C6AL8Z 44274790 IC50 = 9800 nM T85943 CJA7D6 44274792 IC50 = 3000 nM T85943 C4QK7J 44274799 IC50 = 2300 nM T85943 CF81JQ 44274805 IC50 = 500000 nM T85943 CRK9A8 44274807 IC50 = 18500 nM T85943 C9N2RZ 44286529 IC50 = 300 nM T85943 C41JIF 44286666 IC50 = 5500 nM T85943 CSF6T7 44291065 IC50 = 250000 nM T85943 CZFQ76 44291533 IC50 = 27 nM T85943 C4HS3C 44294447 IC50 > 12500 nM T85943 CV98MQ 44299106 IC50 = 2100 nM T85943 C1VNE3 44299107 IC50 = 1000 nM T85943 CXN7A4 44299111 IC50 = 230 nM T85943 C4FBL8 44299118 IC50 = 1200 nM T85943 CRG0B2 44299119 IC50 = 240 nM T85943 CO17YA 44299125 IC50 = 2600 nM T85943 C0M5KC 44299134 IC50 = 600 nM T85943 CW64UF 44299147 IC50 = 300 nM T85943 CS54RJ 44299168 IC50 = 230 nM T85943 C67GTM 44299169 IC50 = 300 nM T85943 CH3J2E 44299176 IC50 = 10 nM T85943 CD36RY 44299191 IC50 = 700 nM T85943 CT0JR5 44299194 IC50 = 200 nM T85943 C27GVO 44299203 IC50 = 70 nM T85943 C9TRU0 44299204 IC50 = 400 nM T85943 C53MIF 44299217 IC50 = 1000 nM T85943 CZQ4W7 44299233 IC50 = 220 nM T85943 CY6WC0 44299236 IC50 = 70 nM T85943 CUR02C 44299252 IC50 = 400 nM T85943 CS0ZN2 44299266 IC50 = 400 nM T85943 CT9OF3 44299268 IC50 = 800 nM T85943 C3RG0C 44299304 IC50 = 70 nM T85943 CLI97F 44299306 IC50 = 200 nM T85943 C59XRM 44299311 IC50 = 150 nM T85943 CJM26I 44299321 IC50 = 50 nM T85943 C9UGL3 44299325 IC50 = 100 nM T85943 CJEZ96 44299338 IC50 = 70 nM T85943 C8XGN5 44299339 IC50 = 40 nM T85943 CHMA85 44299352 IC50 = 300 nM T85943 CNH34G 44299354 IC50 = 30 nM T85943 C65KVU 44299356 IC50 = 2300 nM T85943 C82MSD 44299360 IC50 = 60 nM T85943 C74LKX 44299364 IC50 = 1100 nM T85943 C9W4YN 44299376 IC50 = 700 nM T85943 C4ZBD8 44299385 IC50 = 500 nM T85943 CX0N9E 44299403 IC50 = 10000 nM T85943 CIGR38 44299422 IC50 = 300 nM T85943 CGN5F2 44299425 IC50 = 500 nM T85943 CCH89M 44300026 IC50 = 44000 nM T85943 CV5QH7 44300064 IC50 = 1100 nM T85943 CTJV27 44300144 IC50 = 1800 nM T85943 CVD6B1 44300175 IC50 = 6700 nM T85943 CA2HD0 44300205 IC50 = 4900 nM T85943 CJQ1T0 44300215 IC50 = 5500 nM T85943 CBGM82 44300226 IC50 = 6100 nM T85943 C9FX3G 44300234 IC50 = 9300 nM T85943 CKB2H9 44303538 IC50 = 4.4 nM T85943 CEZF96 44303555 IC50 = 3.8 nM T85943 CA37TL 44303560 IC50 = 4.2 nM T85943 C1CXM5 44303586 IC50 = 2 nM T85943 CXP1C8 44305333 IC50 = 69000 nM T85943 C9VT8P 44307444 IC50 = 133000 nM T85943 C48MLF 44307445 IC50 = 20000 nM T85943 CE78UK 44307458 IC50 = 5000 nM T85943 C63NKT 44307477 IC50 = 29000 nM T85943 CKWS27 44307582 IC50 = 46000 nM T85943 CFHT80 44307583 IC50 = 23000 nM T85943 CMDI19 44307619 IC50 = 164000 nM T85943 C3J7OB 44307626 IC50 = 13000 nM T85943 CV6R3S 44307664 IC50 = 128000 nM T85943 C7GV5F 44307684 IC50 = 873000 nM T85943 C0IE8B 44307685 IC50 = 300 nM T85943 CPN64K 44307686 IC50 = 130 nM T85943 CZEJ78 44307727 IC50 = 400 nM T85943 C0KCL7 44307728 IC50 = 9300 nM T85943 CIY29X 44307740 IC50 = 115000 nM T85943 CV9B6T 44307793 IC50 = 422000 nM T85943 C6N8ME 44307794 IC50 = 1000 nM T85943 C9AOR4 44307795 IC50 = 14200 nM T85943 CT5I2B 44307814 IC50 = 32000 nM T85943 C01UZY 44307844 IC50 = 23000 nM T85943 C7DZ9P 44307845 IC50 = 27000 nM T85943 C5P3QB 44307858 IC50 = 1600 nM T85943 CU7GT2 44307964 IC50 = 1200 nM T85943 C6QV0W 44307989 IC50 = 95000 nM T85943 CMLP98 44308018 IC50 = 1600 nM T85943 CV50HL 44308076 IC50 = 6400 nM T85943 C1L2ID 44308077 IC50 = 18000 nM T85943 CX57AN 44308086 IC50 = 1000 nM T85943 CE35CL 44308217 IC50 = 339000 nM T85943 CEU2W4 44308690 IC50 = 84 nM T85943 CY6ZB5 44308830 IC50 = 150 nM T85943 CQ60AZ 44311887 IC50 = 2800 nM T85943 CM94QU 44311968 IC50 = 3300 nM T85943 C9G3NO 44311969 IC50 = 2700 nM T85943 C9SQU0 44311977 IC50 = 5300 nM T85943 CGQF10 44312058 IC50 = 2000 nM T85943 CQ21ZA 44312059 IC50 = 6900 nM T85943 C43VTG 44312102 IC50 = 2700 nM T85943 CR6D9P 44312116 IC50 = 6500 nM T85943 CF54TL 44312160 IC50 = 4300 nM T85943 CVM42H 44312201 IC50 = 14400 nM T85943 C79XAL 44312222 IC50 = 20000 nM T85943 C9AKW0 44312281 IC50 = 18000 nM T85943 C16XBZ 44312282 IC50 = 10000 nM T85943 C5V8GB 44312283 IC50 = 2700 nM T85943 C5JDT3 44312430 IC50 = 4500 nM T85943 CR24ML 44312445 IC50 = 6700 nM T85943 CO3AR9 44312505 IC50 = 1200 nM T85943 CSAL07 44312506 IC50 = 20000 nM T85943 C3KRV4 44312535 IC50 = 11000 nM T85943 CBNM24 44312579 IC50 = 26000 nM T85943 CJ3PF9 44313929 IC50 > 500000 nM T85943 CUV7K3 44313930 IC50 = 378000 nM T85943 CHK9N3 44313931 IC50 = 3200 nM T85943 CEKR19 44313990 IC50 > 500000 nM T85943 CD5PI9 44313997 IC50 = 2700 nM T85943 C0GH7J 44314372 IC50 = 370000 nM T85943 C5E4GK 44314373 IC50 > 500000 nM T85943 C3YD1G 44314380 IC50 = 35400 nM T85943 CPC68H 44314402 IC50 > 500000 nM T85943 C06JSA 44315296 IC50 = 306000 nM T85943 CY0V9F 44315638 IC50 = 62000 nM T85943 CQER69 44315658 IC50 = 22000 nM T85943 CKLV10 44315679 IC50 = 16000 nM T85943 C5KJX6 44315680 IC50 = 16000 nM T85943 CR2ZL9 44315713 IC50 = 279000 nM T85943 CG6XO0 44315714 IC50 = 89000 nM T85943 C7T9UM 44315734 IC50 = 218000 nM T85943 C1WE6N 44315741 IC50 = 12000 nM T85943 C0BVU8 44315742 IC50 = 25000 nM T85943 CR26JG 44315770 IC50 = 896000 nM T85943 CJ7I4U 44315809 IC50 = 61000 nM T85943 C67LWX 44315810 IC50 = 166000 nM T85943 CXSK19 44315865 IC50 = 2780000 nM T85943 CHM0Z4 44315866 IC50 = 76000 nM T85943 CZN96M 44315880 IC50 = 29000 nM T85943 C9A3DN 44315881 IC50 = 25000 nM T85943 C1HR5W 44315882 IC50 = 24000 nM T85943 CD15ZY 44315883 IC50 = 92000 nM T85943 CW71JX 44315898 IC50 = 384000 nM T85943 C4J7XE 44315899 IC50 = 320000 nM T85943 CZW79B 44315919 IC50 = 14000 nM T85943 CMUR89 44315949 IC50 = 111000 nM T85943 CV91XM 44315960 IC50 = 36000 nM T85943 C1HP8L 44315961 IC50 = 35000 nM T85943 CKN9L1 44315962 IC50 = 33000 nM T85943 C1RGE3 44315963 IC50 = 150 nM T85943 CSO2L9 44315968 IC50 = 65000 nM T85943 CP43UD 44316041 IC50 = 21000 nM T85943 C65NTY 44316297 IC50 = 100000 nM T85943 C6Q8YK 44316404 IC50 = 5000000 nM T85943 CR5KT3 44317894 IC50 = 10 ug.mL-1 T85943 CY6P9K 44318047 IC50 > 100000 nM T85943 CO81DL 44318069 IC50 = 2.5 ug.mL-1 T85943 C0COP5 44318070 IC50 > 20 ug.mL-1 T85943 C4KS5N 44320732 IC50 = 10 nM T85943 CC6YI7 44320769 Ki = 3.2 nM T85943 CXM61A 44321260 Ki = 17 nM T85943 C2FST3 44324647 IC50 = 90 nM T85943 C92TBJ 44324648 IC50 = 500 nM T85943 CI8YR0 44324649 IC50 = 7000 nM T85943 C7JYP4 44324728 IC50 = 54000 nM T85943 CY69SU 44324769 IC50 = 55000 nM T85943 CI93QN 44330124 IC50 = 4000 nM T85943 CCL6N3 44330125 IC50 = 13000 nM T85943 C13ZHT 44330158 IC50 = 7600 nM T85943 CJ5KF3 44330203 IC50 = 9600 nM T85943 CV28HP 44330291 IC50 = 2300 nM T85943 C46QSB 44330307 IC50 = 2700 nM T85943 C8XAZ5 44330511 IC50 = 340 nM T85943 CZNJ34 44330550 IC50 = 290 nM T85943 C6U4LS 44330556 IC50 = 143 nM T85943 CKMN15 44331838 IC50 = 16 nM T85943 CV7XB9 44331839 IC50 = 3.3 nM T85943 C8QKX4 44331973 IC50 > 10000 nM T85943 C5Z6BH 44332009 IC50 = 9.8 nM T85943 C6BX3J 44332079 IC50 > 10000 nM T85943 CX04DQ 44332978 IC50 = 198000 nM T85943 C6IWT8 44334350 IC50 = 310 nM T85943 CDJ4M7 44334410 IC50 = 40 nM T85943 CICU19 44334510 IC50 = 750 nM T85943 C1IGJ8 44334511 IC50 = 1300 nM T85943 C4OC8J 44334512 IC50 = 200 nM T85943 CKPG81 44334515 IC50 = 9810 nM T85943 C0HS9Q 44334516 IC50 = 5230 nM T85943 C9ONY7 44334560 IC50 = 77 nM T85943 C6BC2W 44334685 IC50 = 100 nM T85943 CFW80Z 44334688 IC50 = 15700 nM T85943 C9WG0F 44334742 IC50 = 4 nM T85943 C8LC4R 44334809 IC50 = 48200 nM T85943 C2B9MU 44334854 IC50 = 250 nM T85943 CED5S3 44334867 IC50 = 700 nM T85943 CJV6Y5 44334947 IC50 = 1500 nM T85943 C5KCW0 44335063 IC50 = 120 nM T85943 CR0A1N 44335069 IC50 = 19000 nM T85943 CI26MV 44335070 IC50 = 870 nM T85943 CY82QR 44335071 IC50 = 2500 nM T85943 CD6Q8G 44335105 IC50 = 360 nM T85943 C8BXO3 44335106 IC50 = 40000 nM T85943 C1F4CM 44335113 IC50 = 680 nM T85943 CFM28G 44335153 IC50 = 22000 nM T85943 CLHP54 44335174 IC50 = 60 nM T85943 C1KSW5 44335197 IC50 = 160 nM T85943 CDRP13 44335457 IC50 = 4000 nM T85943 C3IA7S 44335458 IC50 = 40 nM T85943 CLE5C1 44336706 IC50 = 34600 nM T85943 C16GTA 44336731 IC50 = 83200 nM T85943 CPZ75G 44344150 IC50 = 40000 nM T85943 C0KD4U 44346053 IC50 > 10000 nM T85943 C0HZX2 44348186 IC50 = 800 nM T85943 CY7M0E 44351586 IC50 = 1.4 nM T85943 CL5QU9 44352816 IC50 = 160 nM T85943 CRV1T2 44352826 IC50 = 200 nM T85943 CVHA74 44352970 IC50 = 1800 nM T85943 CQ2F5D 44352972 IC50 = 600 nM T85943 C9RUC6 44353122 IC50 = 240 nM T85943 CZ2YC5 44353697 IC50 = 20000 nM T85943 C8NBI3 44353815 IC50 = 237000 nM T85943 C8J1NC 44353827 IC50 = 312000 nM T85943 C8FVG3 44353828 IC50 = 261000 nM T85943 CX6AW4 44356396 IC50 = 3200 nM T85943 CYV2D7 44368815 IC50 > 10000 nM T85943 C2HJ3F 44373834 IC50 = 7900 nM T85943 C8LZ0Q 44381185 IC50 = 10 nM T85943 C6FCU8 44381190 IC50 = 38 nM T85943 C1D2LU 44381191 IC50 = 50 nM T85943 CJZD30 44381192 IC50 = 3 nM T85943 CFQ57C 44381224 IC50 = 79.43 nM T85943 CZ64TC 44381237 IC50 = 1 nM T85943 C5WQY2 44381238 IC50 = 19.95 nM T85943 CM64RL 44381269 IC50 = 3.981 nM T85943 CBKP57 44381381 IC50 = 39.81 nM T85943 CDVX68 44381383 IC50 = 199.53 nM T85943 CZS34I 44381396 IC50 = 400 nM T85943 C2DCJ0 44381398 IC50 = 180 nM T85943 C7I5UF 44381399 IC50 = 50 nM T85943 C6LSB4 44381409 IC50 = 6 nM T85943 CE7H4L 44381435 IC50 = 125.89 nM T85943 CEQ7M0 44381445 IC50 = 47 nM T85943 CP1S0U 44381529 IC50 = 130 nM T85943 CM12OK 44381530 IC50 = 100 nM T85943 C6R1FI 44381547 IC50 = 600 nM T85943 CZ5DL9 44381548 IC50 = 410 nM T85943 C6LC8M 44381556 IC50 = 15 nM T85943 CF8G6M 44381557 IC50 = 35 nM T85943 CCA56B 44381571 IC50 = 84 nM T85943 CS6Z3M 44381575 IC50 = 300 nM T85943 C5Z9MJ 44381580 IC50 = 63.1 nM T85943 CC1IK4 44381584 IC50 = 5 nM T85943 C2FX9T 44381585 IC50 = 15 nM T85943 CFDK49 44381586 IC50 = 5000 nM T85943 CY58LS 44381608 IC50 = 270 nM T85943 CT01OH 44381612 IC50 = 8 nM T85943 C25AJR 44381659 IC50 = 95 nM T85943 CVB7X8 44381660 IC50 = 300 nM T85943 C6DQX7 44381674 IC50 = 5 nM T85943 CBSC06 44381798 IC50 = 24 nM T85943 C25EWD 44381813 IC50 = 130 nM T85943 CBE14A 44381814 IC50 = 350 nM T85943 C32JVZ 44381827 IC50 = 2000 nM T85943 C5M3ZC 44382107 IC50 = 10 nM T85943 C75NGL 44384514 IC50 = 10000 nM T85943 CV0F4D 44384547 IC50 = 63.1 nM T85943 CQF8Y7 44384548 IC50 = 316.23 nM T85943 CI2L9R 44384964 IC50 = 31.62 nM T85943 CC09FT 44384965 IC50 = 31.62 nM T85943 CE9PU7 44385035 IC50 = 5011.87 nM T85943 CQGW07 44385080 IC50 = 199.53 nM T85943 CL4Y9M 44385116 IC50 = 63.1 nM T85943 CFT4H8 44385517 IC50 > 150000 nM T85943 CUI34C 44385739 IC50 = 6309.57 nM T85943 CR81QO 44385763 IC50 = 55000 nM T85943 C13TBV 44385823 IC50 = 88000 nM T85943 C5AE8K 44385824 IC50 > 100000 nM T85943 CLO34G 44386410 IC50 > 150000 nM T85943 CM3A2W 44386411 IC50 > 150000 nM T85943 CO7XC6 44386412 IC50 > 100000 nM T85943 COLU85 44386471 IC50 > 100000 nM T85943 CDXM28 44386472 IC50 > 150000 nM T85943 CSE8N9 44386635 IC50 = 73000 nM T85943 C4YJL1 44386888 IC50 > 100000 nM T85943 CID8J0 44387059 IC50 = 38000 nM T85943 CY7S8D 44390435 IC50 = 2 nM T85943 CK4PS1 44390468 IC50 = 11 nM T85943 CVL94F 44390486 IC50 = 440 nM T85943 C0CAH8 44390498 IC50 = 10 nM T85943 CG6L7O 44390509 IC50 = 37 nM T85943 CY1I7R 44390510 IC50 = 6.6 nM T85943 CWQ90B 44393241 IC50 = 864000 nM T85943 CB58JN 44393258 IC50 = 713000 nM T85943 CU07NW 44393373 IC50 = 396000 nM T85943 CKZY56 44393404 IC50 = 714000 nM T85943 CWOE90 44393412 IC50 = 663000 nM T85943 C4YU9L 44402859 IC50 = 13 nM T85943 C0T1QP 44402860 IC50 = 52 nM T85943 CVD4Q2 44404624 IC50 > 100000 nM T85943 C53MNL 44404626 IC50 > 100000 nM T85943 CL0KQ2 44404627 IC50 > 100000 nM T85943 CZ4VX0 44405504 IC50 = 90000 nM T85943 CRD24A 44405548 IC50 = 5 nM T85943 CD2T6B 44405551 IC50 = 140 nM T85943 COSI79 44405552 IC50 = 5 nM T85943 C5E0NF 44405556 IC50 = 400 nM T85943 C2M7EK 44405584 IC50 = 7 nM T85943 CK84OX 44405585 IC50 < 4 nM T85943 CQ95VK 44405700 IC50 = 15 nM T85943 C4ZN5K 44405706 IC50 < 4 nM T85943 C3NKD4 44405727 IC50 = 350 nM T85943 C1IZU5 44405750 IC50 < 4 nM T85943 C68GPB 44405755 IC50 = 20 nM T85943 CYS5N9 44405756 IC50 = 6 nM T85943 CR32YM 44408182 Ki = 23000 nM T85943 CN84XS 44408186 Ki = 9200 nM T85943 CO8D3Z 44408267 Ki = 12000 nM T85943 CV09DY 44410717 IC50 > 10000 nM T85943 CP3CI1 44410720 IC50 > 10000 nM T85943 C8W7AD 44410723 IC50 > 10000 nM T85943 CAT5X4 44410829 IC50 > 10000 nM T85943 CC6Y5P 44410844 IC50 > 10000 nM T85943 CG34TY 44410851 IC50 > 10000 nM T85943 C41EIA 44410869 IC50 > 10000 nM T85943 CB6AE8 44410948 IC50 > 10000 nM T85943 CXZG12 44410949 IC50 > 10000 nM T85943 CS7IE9 44410953 IC50 > 10000 nM T85943 CA9M4X 44410954 IC50 > 10000 nM T85943 C3SP5H 44410955 IC50 > 10000 nM T85943 C5D6YP 44410956 IC50 > 10000 nM T85943 C5W1VC 44410959 IC50 > 10000 nM T85943 CM1C2G 44410960 IC50 > 10000 nM T85943 CVSI80 44411048 IC50 > 10000 nM T85943 CN72BR 44411161 IC50 > 10000 nM T85943 C4AW0O 44411183 IC50 > 10000 nM T85943 C54HEG 44412002 IC50 > 700000 nM T85943 C8E7RS 44412008 IC50 = 280 nM T85943 CJ5V1R 44412134 IC50 > 700000 nM T85943 C7UZ8F 44414044 IC50 = 120 nM T85943 CH6QD2 44414076 IC50 = 15 nM T85943 CHG8W7 44414077 IC50 = 9.9 nM T85943 C0RA6X 44414100 IC50 = 9 nM T85943 COM36D 44414101 IC50 = 5.3 nM T85943 C83TGR 44414121 IC50 = 4.3 nM T85943 CJY27H 44414122 IC50 = 4.2 nM T85943 CNM32J 44414123 IC50 = 22 nM T85943 C6YQ4I 44414139 IC50 = 2700 nM T85943 CHV86W 44414158 IC50 = 18 nM T85943 CPNR25 44414160 IC50 = 150 nM T85943 CLN1F8 44414175 IC50 = 87 nM T85943 CH8BO1 44414190 IC50 = 4.9 nM T85943 CNX21O 44414205 IC50 = 120 nM T85943 C93JTL 44414301 IC50 = 29 nM T85943 C3Z7VW 44414581 IC50 = 104 nM T85943 C8ED2X 44414624 IC50 = 273 nM T85943 C8G5YN 44415111 IC50 = 7 nM T85943 CHJ7T1 44415158 IC50 = 1 nM T85943 C5TQ4F 44415291 IC50 = 6 nM T85943 CLQ8W9 44417523 IC50 = 3 nM T85943 C2LDT6 44417577 IC50 = 55 nM T85943 C7F8GP 44417581 IC50 = 9.5 nM T85943 CS7AK6 44419368 IC50 = 130 nM T85943 CU5MK2 44419371 IC50 > 50000 nM T85943 COAW26 44419397 IC50 = 480 nM T85943 C1Q2JV 44419398 IC50 = 128 nM T85943 CHJ9U5 44419413 IC50 > 50000 nM T85943 C0A5WH 44419420 IC50 = 1800 nM T85943 C3J9IU 44419423 IC50 = 32 nM T85943 CQ9OK4 44419428 IC50 = 21 nM T85943 CE1J7V 44419429 IC50 = 36 nM T85943 C48JXM 44419431 IC50 = 40 nM T85943 CIK43E 44419432 IC50 = 41 nM T85943 C8IZ7D 44419438 IC50 = 9 nM T85943 C2Z3FW 44419440 IC50 = 26 nM T85943 CM6GY0 44419442 IC50 = 320 nM T85943 C5P4VY 44419450 IC50 = 137 nM T85943 CF3ZG4 44419454 IC50 = 240 nM T85943 CE7DB6 44419466 IC50 = 140 nM T85943 C9X5DJ 44421363 IC50 = 21 nM T85943 CWC9T1 44421365 IC50 > 10000 nM T85943 CU39RW 44421388 IC50 = 240 nM T85943 C8HOG7 44422489 IC50 = 13 nM T85943 CG9YW5 44422500 IC50 = 42 nM T85943 C5LK7N 44422501 IC50 = 490 nM T85943 CCBY03 44422511 IC50 = 38 nM T85943 C4RKD6 44422512 IC50 = 693 nM T85943 C65NOR 44422516 IC50 = 1000000 nM T85943 CH6EJ2 44422517 IC50 = 15 nM T85943 CB7LE6 44422520 IC50 = 260 nM T85943 CJSV42 44422521 IC50 = 3700 nM T85943 CEV0F3 44422549 IC50 = 235 nM T85943 C6V5ID 44422550 IC50 = 52 nM T85943 CBE5L3 44422555 IC50 = 108 nM T85943 CTF7N8 44422556 IC50 = 12 nM T85943 C72OSJ 44422563 IC50 = 59 nM T85943 C04PHR 44422564 IC50 = 145 nM T85943 CQ9CU6 44422569 IC50 = 42 nM T85943 CH4L7R 44422570 IC50 = 37 nM T85943 CIQC36 44422581 IC50 = 55 nM T85943 CN7GM6 44422617 IC50 = 235 nM T85943 C3ATF6 44422621 IC50 = 23 nM T85943 CY9PW1 44422622 IC50 = 3300 nM T85943 CPSU79 44422629 IC50 = 235 nM T85943 CW8A6F 44422630 IC50 = 19 nM T85943 C9Z7NE 44425253 IC50 = 505 nM T85943 C4HTU1 44425257 IC50 = 1200 nM T85943 C0MFI1 44425259 IC50 = 204 nM T85943 C6A4ID 44425260 IC50 = 207 nM T85943 CRC92J 44425261 IC50 = 1500 nM T85943 CJ25XD 44425262 IC50 = 1800 nM T85943 C67BFA 44425263 IC50 = 30 nM T85943 C9YZ5V 44425264 IC50 > 10000 nM T85943 CCER34 44425265 IC50 = 12 nM T85943 CLE93Z 44425266 IC50 = 51 nM T85943 CAY37H 44425267 IC50 = 282 nM T85943 CO36YB 44425268 IC50 = 353 nM T85943 CDE3L4 44425269 IC50 = 631 nM T85943 C1L5QJ 44425270 IC50 = 2900 nM T85943 C93JFH 44425275 IC50 = 11 nM T85943 C4FZW3 44425278 IC50 = 315 nM T85943 CF9U4X 44425280 IC50 > 10000 nM T85943 C0D3SP 44425282 IC50 > 10000 nM T85943 CB75SQ 44425284 IC50 = 10 nM T85943 CHW46S 44425285 IC50 = 67 nM T85943 C3D2ZL 44425287 IC50 = 20 nM T85943 CH4N0C 44425289 IC50 = 92 nM T85943 C9VI3O 44425291 IC50 = 72 nM T85943 C8M9TC 44425295 IC50 = 33 nM T85943 CM0F3I 44425296 IC50 = 40 nM T85943 C85BYK 44425297 IC50 = 36 nM T85943 CV23XW 44425298 IC50 = 39 nM T85943 C6BY7F 44425299 IC50 = 15 nM T85943 C9V0ZI 44425300 IC50 = 13 nM T85943 CN8S5L 44425301 IC50 = 16 nM T85943 CN9QL8 44425302 IC50 = 18 nM T85943 CKQ42L 44425303 IC50 = 6.4 nM T85943 CO8BX5 44425311 IC50 = 10 nM T85943 C4ANK9 44425312 IC50 = 10 nM T85943 CQXB26 44425313 IC50 = 14 nM T85943 CJ09ND 44425314 IC50 = 21 nM T85943 CETQ79 44427518 IC50 > 50000 nM T85943 COPG94 44427519 IC50 > 10000 nM T85943 CC2T8I 44435575 Ki = 25000 nM T85943 C5ZKI8 44435586 Ki = 1710 nM T85943 CO3LT4 44439198 IC50 = 11 nM T85943 C2RVA8 44439199 IC50 = 4.9 nM T85943 C8Q4RH 44439200 IC50 = 4.1 nM T85943 CX79TF 44439201 IC50 = 5.4 nM T85943 CUE35S 44439202 IC50 = 28 nM T85943 C7R2JB 44439203 IC50 = 230 nM T85943 C2M4ZC 44439204 IC50 = 8.7 nM T85943 C6J4WX 44439205 IC50 = 4.1 nM T85943 C0QG4D 44439207 IC50 = 21 nM T85943 CZRG28 44439212 IC50 = 220 nM T85943 CGV37F 44440254 IC50 = 43311 nM T85943 C5JUV3 44440256 IC50 > 50000 nM T85943 CFB56S 44440259 IC50 > 50000 nM T85943 CEW9G2 44440261 IC50 > 50000 nM T85943 C5R4QE 44442729 Ki = 150 nM T85943 CGC76I 44442730 Ki = 170 nM T85943 CJM6N5 44442731 Ki = 210 nM T85943 CH2FS6 44442732 Ki = 330 nM T85943 CZ7FC6 44442733 Ki > 10000 nM T85943 C6PNZ4 44442734 Ki > 10000 nM T85943 C8N1EQ 44442735 Ki > 10000 nM T85943 C26EVP 44442736 Ki = 49 nM T85943 C0S6PN 44442737 Ki = 110 nM T85943 CAZ5O7 44442738 Ki = 45 nM T85943 CM9XW1 44442739 Ki > 10000 nM T85943 CFOH51 44442740 Ki = 280 nM T85943 CX10DZ 44442742 Ki = 86 nM T85943 CN12IA 44442744 Ki = 570 nM T85943 C0DOP6 44442745 Ki = 140 nM T85943 C1L6MG 44444041 IC50 = 3.6 nM T85943 C4YMI9 44447890 IC50 = 43 nM T85943 CR65PM 44447895 IC50 = 14 nM T85943 CSA12W 44450544 IC50 > 400000000 nM T85943 CSG8K7 44452043 IC50 = 100 nM T85943 CGT37L 44452045 IC50 = 5 nM T85943 CQ4T3N 44452085 IC50 = 12 nM T85943 C8WY2S 44452121 IC50 = 25 nM T85943 C1DH0Z 44452147 IC50 = 8 nM T85943 CK4T8L 44452148 IC50 = 93 nM T85943 CWA9S7 44452173 IC50 = 68 nM T85943 CJ1P5Q 44452174 IC50 = 41 nM T85943 C65YLS 44452200 IC50 = 1210 nM T85943 CZ57PB 44452201 IC50 = 432 nM T85943 CL8E6C 44452225 IC50 = 9200 nM T85943 CAPE54 44452226 IC50 = 3480 nM T85943 C0LPT5 44452252 IC50 = 6690 nM T85943 CBU8P5 44454498 Ki = 195 nM T85943 C0ZL8E 44454721 Ki = 272 nM T85943 C3RY8Z 44454722 Ki = 169 nM T85943 C2KJO6 44454776 Ki = 170 nM T85943 CA2JO0 44454803 Ki = 199 nM T85943 CH64KP 44454904 Ki = 165 nM T85943 C6CQJ0 44454939 Ki = 219 nM T85943 C8IZ1S 44459512 IC50 = 1700 nM T85943 CQDS15 44459528 IC50 = 2300 nM T85943 C46MXA 44459547 IC50 = 1800 nM T85943 CS1P8H 44459548 IC50 = 2040 nM T85943 CAV83X 44459562 IC50 = 2100000 nM T85943 CSBU10 44459581 IC50 = 2160 nM T85943 CR3O4A 44459585 IC50 = 4000000 nM T85943 CBZ54E 44459587 IC50 = 3900000 nM T85943 CDC20A 44459602 IC50 = 3600000 nM T85943 CH2MB0 44459619 IC50 = 3300000 nM T85943 CEZY71 44459644 IC50 = 334 nM T85943 C3NX1Q 44459658 IC50 = 1200000 nM T85943 CJ27KA 44459670 IC50 = 150 nM T85943 CYXJ43 44459671 IC50 = 1300 nM T85943 CO9HE5 44459688 IC50 = 315 nM T85943 C2AC0U 44459689 IC50 = 26 nM T85943 C6Y5UT 44459690 IC50 = 87 nM T85943 C53BRW 44459721 IC50 = 58 nM T85943 C89CKB 44459723 IC50 = 15200 nM T85943 C2R8QH 44459724 IC50 = 2110 nM T85943 CTW28U 44459744 IC50 = 300000 nM T85943 C0SF6A 44459789 IC50 = 3500000 nM T85943 CUR73W 44459790 IC50 = 1500 nM T85943 CA6SD1 44459791 IC50 = 11900 nM T85943 C28LMK 44459792 IC50 = 10400 nM T85943 CWM2I1 44459805 IC50 = 3200000 nM T85943 C5FC2Q 44459806 IC50 = 2460 nM T85943 CM3EA7 44459859 IC50 = 4000000 nM T85943 C61WOQ 44459904 IC50 >> 5000000 nM T85943 CD8WC3 44459920 IC50 = 600000 nM T85943 C7X2SW 44459923 IC50 = 280 nM T85943 C71EPS 44460198 IC50 = 12.5 ug.mL-1 T85943 CLBX75 44460201 IC50 = 1.8 ug.mL-1 T85943 C9O1DQ 44460220 IC50 = 1.3 ug.mL-1 T85943 C3PAD4 44460222 IC50 > 10 ug.mL-1 T85943 CLNZ91 44460237 IC50 = 3.2 ug.mL-1 T85943 C9Z8XJ 44460238 IC50 > 10 ug.mL-1 T85943 CH9F0N 44460247 IC50 = 1.3 ug.mL-1 T85943 CV1Q0D 44460258 IC50 = 1.9 ug.mL-1 T85943 C4RGQ0 44461745 IC50 > 10000 nM T85943 CWM1I0 44461758 IC50 = 5.3 nM T85943 CJ3QZ6 44462200 IC50 = 460 nM T85943 CV9Z6W 44517648 IC50 < 0.46 nM T85943 CYH6P3 44520205 IC50 > 10000 nM T85943 C4WRN5 44541014 IC50 = 50000 nM T85943 C3VRO9 44557921 IC50 > 10000 nM T85943 CF16QB 44560451 IC50 = 1210 nM T85943 C0U8DH 44560546 IC50 = 3760 nM T85943 CQL6U3 44561590 IC50 = 1.78 nM T85943 CFS16E 44561591 IC50 = 6.58 nM T85943 CCVU76 44561592 IC50 = 31.8 nM T85943 C4QBE6 44561593 IC50 = 376 nM T85943 CEF4G0 44561735 IC50 = 126 nM T85943 CR87GD 44561736 IC50 = 198 nM T85943 CA25TK 44561737 IC50 = 17 nM T85943 C8TRZ9 44561787 IC50 = 3.74 nM T85943 C7YK5F 44561788 IC50 = 1.43 nM T85943 CDK0X8 44561828 IC50 < 0.23 nM T85943 C38YGU 44561829 IC50 < 0.23 nM T85943 C28NDO 44561830 IC50 < 0.46 nM T85943 C4C6VA 44561831 IC50 < 0.46 nM T85943 CJ73WK 44561866 IC50 < 0.46 nM T85943 CMKB42 44561867 IC50 < 0.46 nM T85943 C1TQ2I 44561868 IC50 < 0.46 nM T85943 C6MA5F 44561869 IC50 < 0.46 nM T85943 CDVC07 44561908 IC50 = 1.29 nM T85943 CLB68G 44561909 IC50 < 0.46 nM T85943 C3Q0DX 44564789 IC50 = 1500 nM T85943 CP40XB 44564790 IC50 > 10000 nM T85943 C35NTB 44564791 IC50 = 6400 nM T85943 CJY83G 44564817 IC50 = 2100 nM T85943 CLK98G 44564818 IC50 > 10000 nM T85943 CF2D1K 44564819 IC50 > 10000 nM T85943 C3CQ9K 44564820 IC50 > 10000 nM T85943 CI8V2L 44564821 IC50 > 10000 nM T85943 C9PO7J 44564860 IC50 > 10000 nM T85943 C16FJW 44564861 IC50 > 10000 nM T85943 C8AMX5 44564862 IC50 = 630 nM T85943 CTR59U 44564863 IC50 > 10000 nM T85943 C9EY4C 44564864 IC50 = 500 nM T85943 CG5Z7T 44564910 IC50 = 700 nM T85943 CU9O4C 44564911 IC50 = 300 nM T85943 CXZ15S 44564954 IC50 > 10000 nM T85943 CZ78WJ 44564955 IC50 = 3000 nM T85943 CJ1X9V 44565013 IC50 = 190 nM T85943 CN2Q3D 44565014 IC50 = 960 nM T85943 CM2GN3 44565015 IC50 > 10000 nM T85943 C6RV9I 44565016 IC50 = 1100 nM T85943 CSZU30 44565566 IC50 = 19.95 nM T85943 C1UN7I 44565567 IC50 = 7.943 nM T85943 C8FB0L 44565568 IC50 = 158.49 nM T85943 CG07MP 44565569 IC50 = 39.81 nM T85943 CQVN71 44565650 IC50 = 125.89 nM T85943 C34IFY 44565651 IC50 = 39.81 nM T85943 CC5LZ3 44565675 IC50 = 5011.87 nM T85943 C2L5IB 44565676 IC50 = 316.23 nM T85943 CZD9U4 44565677 IC50 = 15.85 nM T85943 CP5OF0 44565687 IC50 = 5.012 nM T85943 C7AMV5 44565688 IC50 = 1995.26 nM T85943 C73HDS 44565689 IC50 = 316.23 nM T85943 CSQE94 44565690 IC50 = 125.89 nM T85943 C1HPC3 44565691 IC50 = 50.12 nM T85943 C5N4CU 44565706 IC50 = 398.11 nM T85943 C58UTE 44565707 IC50 = 31.62 nM T85943 CZO20U 44565708 IC50 = 100 nM T85943 C6UAO3 44565709 IC50 = 630.96 nM T85943 CD6VS7 44565726 IC50 = 125.89 nM T85943 C1UFS0 44565727 IC50 = 25.12 nM T85943 CIEC59 44565728 IC50 = 316.23 nM T85943 CHRC09 44565729 IC50 = 100 nM T85943 CW4IZ8 44565793 IC50 = 6309.57 nM T85943 C1SLZ2 44565813 Ki = 3981.07 nM T85943 CG4D6Z 44565814 IC50 = 501.19 nM T85943 C4LY2T 44565815 IC50 = 316.23 nM T85943 CB49VN 44565833 IC50 = 50.12 nM T85943 CO3ES1 44565855 IC50 = 251.19 nM T85943 CW04KX 44565856 IC50 = 501.19 nM T85943 C4F7IL 44565857 IC50 = 5011.87 nM T85943 CN64AE 44565858 IC50 = 39.81 nM T85943 CO53WH 44565859 IC50 = 19.95 nM T85943 CF50OG 44565860 IC50 = 10 nM T85943 C7MER3 44565861 IC50 = 0.3162 nM T85943 C7OBC1 44565875 IC50 = 2511.89 nM T85943 CUY3K2 44565876 IC50 = 3.162 nM T85943 CK9N7B 44565877 IC50 = 0.3162 nM T85943 CDUC85 44565878 IC50 = 19.95 nM T85943 C2QSK9 44565879 IC50 = 19.95 nM T85943 C3HW7L 44570553 IC50 > 30000 nM T85943 C17PVE 44570554 IC50 = 4000 nM T85943 CLOY92 44570599 IC50 = 100 nM T85943 CK06LT 44570600 IC50 = 3000 nM T85943 CJY8S0 44570884 IC50 > 5000 nM T85943 CCL85F 44575073 IC50 > 50000 nM T85943 CJX06P 44575126 IC50 > 50000 nM T85943 CE8FC7 44575127 IC50 > 50000 nM T85943 CXD9B4 44578561 IC50 = 1800 nM T85943 C5SCQ9 44582755 IC50 = 300 nM T85943 CQL93I 44586518 IC50 = 75.9 nM T85943 CAM3T1 44586519 IC50 = 172 nM T85943 C5HQ0C 44586520 IC50 = 209 nM T85943 C1B9LY 44586521 IC50 = 646 nM T85943 CG17XL 44586569 IC50 = 111 nM T85943 C9Y4TF 44586570 IC50 > 1000 nM T85943 CIU7V1 44586571 IC50 = 186 nM T85943 CWP8B5 44586572 IC50 = 178 nM T85943 C9G1JL 44586612 IC50 = 371 nM T85943 CJK4W0 44586613 IC50 > 1000 nM T85943 C4WYU6 44586614 IC50 = 9.23 nM T85943 C2O9TP 44586615 IC50 = 133 nM T85943 CA5UF3 44589514 Ki = 3500 nM T85943 C3KLD1 44589515 Ki = 4000 nM T85943 C7A0UX 44589516 Ki = 3700 nM T85943 CYK07V 44589517 Ki = 1800 nM T85943 CS1V3A 44589852 IC50 = 81.1 nM T85943 CSI36R 44589853 IC50 = 129 nM T85943 C2KT4X 44589904 IC50 = 53.4 nM T85943 CH4T0X 44589905 IC50 = 36.6 nM T85943 CK6V1D 44589906 IC50 = 42 nM T85943 CUOM53 44589964 IC50 = 143 nM T85943 C8THB4 44589965 IC50 = 159 nM T85943 CMKO67 44589966 IC50 = 20.7 nM T85943 C89COX 44590149 Ki = 1833 nM T85943 C2BQ4M 44590150 Ki = 991 nM T85943 C6NB9K 44590204 Ki = 348 nM T85943 CQ0NU8 44590205 Ki = 2230 nM T85943 C2PX5O 44593468 Ki = 153 nM T85943 CZ20KC 44593469 Ki = 3500 nM T85943 CM3T7B 44593470 Ki = 3500 nM T85943 CD2FE4 44593471 Ki = 2030 nM T85943 CS8GE3 44593472 Ki = 1357 nM T85943 CKM4H0 44593475 Ki > 3330 nM T85943 C28QLM 44605035 IC50 > 50000 nM T85943 C75XHS 44605037 IC50 > 50000 nM T85943 CJ2L1M 44820629 IC50 = 48 nM T85943 CP2YM3 45103907 IC50 = 1900 nM T85943 COE8U0 45267045 IC50 = 90000 nM T85943 CPO6K5 45271266 Ki = 796 nM T85943 CZC5V0 45272013 Ki = 4000 nM T85943 CC95PQ 45375865 IC50 = 220 nM T85943 CEOQ27 45375866 IC50 > 50000 nM T85943 C6E2SC 45482700 IC50 > 10000 nM T85943 CZXH74 45482750 IC50 > 10000 nM T85943 CS41VI 45486589 IC50 = 5.1 nM T85943 C6YUM9 45486590 IC50 = 12 nM T85943 C7C3KP 45486594 IC50 = 96 nM T85943 C69ABL 45486610 IC50 = 130 nM T85943 C65TAS 45486623 IC50 = 1.8 nM T85943 CS5U2D 45486634 IC50 = 3.9 nM T85943 CJC6F2 45486640 IC50 = 360 nM T85943 CA06GW 45487959 IC50 = 213 nM T85943 CUMF37 45487992 IC50 = 9.2 nM T85943 CFE79C 45487997 IC50 = 30 nM T85943 C96BNW 46179972 IC50 = 5 nM T85943 CUA97D 46209401 IC50 > 10000 nM T85943 CF57GK 46215462 IC50 = 37 nM T85943 CZBL95 46220496 IC50 = 274 nM T85943 CY3HW5 46224684 IC50 = 6100 nM T85943 C1J6GR 46224908 IC50 = 23 nM T85943 CYT37A 46232443 IC50 = 22000 nM T85943 CG5K2H 46232509 IC50 = 20000 nM T85943 CA98UN 46232510 IC50 > 50000 nM T85943 CPK7Z8 46232511 IC50 > 50000 nM T85943 C8E4RB 46232512 IC50 > 50000 nM T85943 CZ52WR 46232513 IC50 > 50000 nM T85943 CAG90T 46232552 IC50 > 50000 nM T85943 C1O4DG 46232553 IC50 = 46000 nM T85943 CSHX24 46232554 IC50 > 50000 nM T85943 CUE6J3 46742603 IC50 > 100000 nM T85943 CI9SK3 46742606 IC50 = 139000 nM T85943 C0QOJ6 46844437 Ki = 100 nM T85943 CQW97N 46846072 IC50 = 130 nM T85943 C8Q5MT 46861577 IC50 = 2000 nM T85943 C4X3SZ 46861861 IC50 = 78 nM T85943 C91AFI 46861862 IC50 = 2.5 nM T85943 C7H4YM 46865419 IC50 > 10000 nM T85943 C9LI2B 46866423 IC50 = 324 nM T85943 CP68SD 46866425 IC50 = 513 nM T85943 CO3P0J 46866604 IC50 < 50000 nM T85943 CX43UQ 46871756 IC50 = 642 nM T85943 CQB16A 46872415 Ki > 4000 nM T85943 CLS29B 46872626 IC50 > 10000 nM T85943 CRS61F 46879438 IC50 > 10000 nM T85943 C27JEF 46879439 IC50 = 1268 nM T85943 CF0T8P 46879440 IC50 = 1065 nM T85943 C12RMW 46879441 IC50 = 1537 nM T85943 CH2D7N 46879442 IC50 = 1409 nM T85943 CI6OD8 46879443 IC50 = 556 nM T85943 C7YD4Q 46879444 IC50 = 458 nM T85943 C8MN5Q 46879445 IC50 = 364 nM T85943 CX6SW2 46879446 IC50 = 1223 nM T85943 CNF3V6 46879447 IC50 > 2500 nM T85943 CW46VY 46879448 IC50 = 117 nM T85943 CLK6X3 46879907 IC50 = 530 nM T85943 CRPU47 46879908 IC50 = 56 nM T85943 C1TIE9 46880013 IC50 > 10000 nM T85943 C2A8KO 46880066 IC50 = 1288 nM T85943 CBRP80 46880067 IC50 = 1322 nM T85943 C3FY2B 46880068 IC50 = 1661 nM T85943 CX89TY 46880069 IC50 = 139 nM T85943 CB0XY1 46880070 IC50 = 165 nM T85943 CUD81V 46880071 IC50 = 903 nM T85943 CZP58Q 46880072 IC50 = 739 nM T85943 CC8OF9 46880073 IC50 = 524 nM T85943 CF41HG 46880098 IC50 = 606 nM T85943 C6O2YG 46880099 IC50 = 7173 nM T85943 CI78DM 46880100 IC50 = 21 nM T85943 CU04ZK 46880101 IC50 = 202 nM T85943 C4E0MF 46880133 IC50 > 10000 nM T85943 COJ16A 46880134 IC50 = 5375 nM T85943 C71MGJ 46880135 IC50 > 10000 nM T85943 CJOM49 46880136 IC50 = 675 nM T85943 C3R6TL 46880213 IC50 = 4389 nM T85943 CT8BQ4 46880214 IC50 = 6168 nM T85943 C0JTO4 46880215 IC50 = 7613 nM T85943 CAFN49 46880216 IC50 > 10000 nM T85943 C2O8RZ 46886323 IC50 = 310 nM T85943 CFZG89 46888909 IC50 = 280 nM T85943 CI2KA3 46888910 IC50 = 2.2 nM T85943 C82CYI 46888911 IC50 = 2.2 nM T85943 CJ52NV 46888912 IC50 = 2.4 nM T85943 CLH6K1 46888976 IC50 = 3 nM T85943 C8A3PW 46889002 IC50 = 1.7 nM T85943 CXMI58 46889003 IC50 = 260 nM T85943 CT5IB1 46889004 IC50 = 4.8 nM T85943 C8LF3J 46889005 IC50 = 5.4 nM T85943 CC02ON 46889031 IC50 = 290 nM T85943 C9FZ4U 46889032 IC50 = 130 nM T85943 CV2DI3 46889033 IC50 = 15 nM T85943 CKCF96 46889034 IC50 = 2800 nM T85943 CV6LB1 46889053 IC50 = 340 nM T85943 CGAR69 46889054 IC50 = 1200 nM T85943 C1YS5A 46890918 IC50 > 1000 nM T85943 CJ5S3N 46890968 IC50 = 135 nM T85943 CAGE32 46890969 IC50 > 1000 nM T85943 C3A7BP 46890970 IC50 = 1706 nM T85943 CTV73J 46890971 IC50 = 688 nM T85943 CUX9B4 46891024 IC50 = 1000 nM T85943 CG35WP 46891025 IC50 = 227 nM T85943 C3FBH0 46891026 IC50 = 554 nM T85943 CYOU90 46891080 IC50 = 142 nM T85943 CJ16KH 46891081 IC50 = 1000 nM T85943 C7DOF4 46891082 IC50 = 394 nM T85943 CM14YO 46891147 IC50 = 143 nM T85943 CRPL41 46891148 IC50 = 497 nM T85943 C6FJ7G 46891184 IC50 > 1000 nM T85943 C1B2UZ 46891185 IC50 > 1000 nM T85943 CYM5B2 46891226 IC50 > 1000 nM T85943 C2DZE0 46891227 IC50 > 1000 nM T85943 C1W0JX 46891228 IC50 = 762 nM T85943 CI3VZ0 46891275 IC50 > 1000 nM T85943 C0WYM1 46898022 IC50 = 20 nM T85943 CL0O4U 46911726 Ki = 26 nM T85943 C60GAV 46929544 IC50 = 5750 nM T85943 C68MSY 46938699 IC50 = 680 nM T85943 C64IQW 49799035 IC50 = 340 nM T85943 C2BOD5 49799036 IC50 = 260 nM T85943 CNYS09 49799037 IC50 = 340 nM T85943 C0INW7 49799038 IC50 = 1220 nM T85943 CT56HG 49799073 IC50 = 120 nM T85943 CI95GE 49799074 IC50 = 2010 nM T85943 C47KVD 49799075 IC50 = 1590 nM T85943 CUR93J 49799132 IC50 = 650 nM T85943 CM8J0V 49799133 IC50 = 3140 nM T85943 CKP38B 49799178 IC50 = 100 nM T85943 CJ0X9M 49799179 IC50 = 2200 nM T85943 C86HTO 49799180 IC50 = 1050 nM T85943 C1W7YX 49799181 IC50 = 750 nM T85943 C0RGZ8 49799182 IC50 = 130 nM T85943 CN3Y0A 49799214 IC50 > 10000 nM T85943 CJT2C7 49799246 IC50 = 2430 nM T85943 CLK89M 49799247 IC50 = 2420 nM T85943 CV2TB6 49799248 IC50 = 1210 nM T85943 CY9L3I 49799284 IC50 > 10000 nM T85943 CTDW23 49799379 IC50 = 1330 nM T85943 C9B2EV 49799380 IC50 = 1200 nM T85943 C9Q3UO 49799413 IC50 = 2550 nM T85943 CUE29W 49799414 IC50 = 690 nM T85943 CZ4M7C 49799415 IC50 = 780 nM T85943 C5Z2QM 49799434 IC50 = 930 nM T85943 C1EUI9 49799435 IC50 = 830 nM T85943 C62TRB 49799436 IC50 = 340 nM T85943 C6FTC1 49799437 IC50 = 450 nM T85943 CZ53BX 49799438 IC50 = 390 nM T85943 C6CA5J 49799464 IC50 = 1180 nM T85943 CQ1GY5 49799465 IC50 = 130 nM T85943 CEI8Q3 49799502 IC50 = 1760 nM T85943 C9PH0Z 49799503 IC50 = 1400 nM T85943 CE4KQ2 49799504 IC50 = 950 nM T85943 C0TJE7 49799505 IC50 = 1820 nM T85943 CNL8F1 49799533 IC50 > 10000 nM T85943 C4RS5K 49799534 IC50 > 10000 nM T85943 C80SQD 49799535 IC50 > 10000 nM T85943 CHSF07 49806372 IC50 > 1000 nM T85943 C5ME3S 49806721 IC50 > 50000 nM T85943 C2N9UP 49843809 IC50 = 41600 nM T85943 C9OWY0 49850406 Ki = 650 nM T85943 CG32IB 49850407 Ki = 770 nM T85943 C8EOD9 49850435 Ki = 200 nM T85943 CX61ON 49865963 IC50 = 208 nM T85943 CF4V7Z 49867019 IC50 = 65 nM T85943 CQ3KU9 50899556 IC50 = 61 nM T85943 C90ANW 50939489 IC50 = 3400 nM T85943 C6XYT1 50941838 IC50 = 33900 nM T85943 CS9G6E 50997096 IC50 > 10000 nM T85943 CY50QZ 51003413 IC50 = 5600 nM T85943 C4OSU5 51003414 IC50 = 17400 nM T85943 CK0RE5 51003422 IC50 = 9100 nM T85943 C43HGW 51003423 IC50 = 29600 nM T85943 C46STW 51346068 Ki = 160000 nM T85943 CH1WR3 52914084 IC50 = 88 nM T85943 C13MUQ 52914647 IC50 = 544 nM T85943 CROJ51 52920524 IC50 = 246 nM T85943 CTX8B2 52920590 IC50 = 32 nM T85943 C9E5PQ 52920591 IC50 = 40 nM T85943 C1VML8 52936434 Ki = 1800 nM T85943 CU1T5C 52936530 Ki = 140 nM T85943 CK69ML 52936531 Ki = 40 nM T85943 CCT6B9 52936532 Ki = 1200 nM T85943 CC7SE4 52936533 Ki = 220 nM T85943 CA93FM 52936534 Ki = 590 nM T85943 C9KO7D 52936535 Ki = 590 nM T85943 CEQN27 52936621 Ki = 120 nM T85943 C2A6MX 52936622 Ki = 280 nM T85943 CBH0K9 52936623 Ki = 300 nM T85943 CKF2D5 52936624 Ki = 480 nM T85943 CM24LF 52938983 IC50 = 4.79 nM T85943 CU1P2L 52940797 IC50 = 9800 nM T85943 C3LB5V 52941849 IC50 = 3200 nM T85943 CDHJ08 52942235 IC50 = 15000 nM T85943 C1XEV2 52943394 IC50 = 144 nM T85943 CW2X5E 52944268 IC50 = 96 nM T85943 CWPC54 52945348 IC50 = 1200 nM T85943 C4NLX7 52945630 IC50 = 2000 nM T85943 C9PX2J 52945752 IC50 = 3300 nM T85943 CL4ED3 52945753 IC50 = 21 nM T85943 CXD6T8 52945845 IC50 = 3400 nM T85943 CIR3Q0 52947964 IC50 = 8200 nM T85943 CHJS47 52951432 Ki = 7600 nM T85943 CY6JF8 52951435 Ki = 740 nM T85943 CE03RQ 52951437 Ki = 3000 nM T85943 C4LDA0 52951544 Ki = 2400 nM T85943 C9UH8Q 52951545 Ki = 3800 nM T85943 C0LTS2 52951546 Ki = 2900 nM T85943 C2MVU5 52951547 Ki = 1200 nM T85943 CY7W0Z 52951664 Ki = 190 nM T85943 CBI6V7 52951665 Ki = 210 nM T85943 C93XNY 52951666 Ki = 3000 nM T85943 CJ7UC0 52951667 Ki = 8300 nM T85943 CE5YZ0 52951668 Ki = 3900 nM T85943 C9OX0Z 52951669 Ki = 4800 nM T85943 C09SDH 53257410 IC50 > 10000 nM T85943 CU95KZ 53316738 Ki = 1760 nM T85943 C1LK0N 53317214 IC50 > 75000 nM T85943 CS7IO3 53317355 IC50 = 72800 nM T85943 CC1FT2 53317356 IC50 > 150000 nM T85943 CE0PS8 53317358 IC50 = 89500 nM T85943 CB24XW 53317359 IC50 = 32500 nM T85943 CFJ78X 53317360 IC50 > 150000 nM T85943 C4XTJ8 53317361 IC50 = 43200 nM T85943 CYXG92 53317690 IC50 > 75000 nM T85943 CX51DG 53318638 IC50 > 100000 nM T85943 C46JSW 53318639 IC50 > 100000 nM T85943 C97HOV 53318640 IC50 > 100000 nM T85943 CKL6Q8 53318898 IC50 > 75000 nM T85943 C50AFD 53319964 IC50 = 81000 nM T85943 CQL6G9 53320214 IC50 = 16400 nM T85943 C7I8AY 53321267 IC50 = 49800 nM T85943 C4BC7G 53321269 IC50 = 62100 nM T85943 C7EUI1 53321272 IC50 = 66100 nM T85943 C9FYE0 53321527 IC50 = 6200 nM T85943 CETZ20 53322857 IC50 > 75000 nM T85943 C9J7FT 53322858 IC50 > 75000 nM T85943 CD74XV 53322859 IC50 > 75000 nM T85943 C5J8UF 53322860 IC50 > 75000 nM T85943 C6XBM0 53322861 IC50 > 75000 nM T85943 CY19KR 53323927 IC50 > 150000 nM T85943 CJH0A1 53323928 IC50 > 150000 nM T85943 CWE4C2 53324181 IC50 > 75000 nM T85943 CS5D3L 53324182 IC50 = 23100 nM T85943 CZ7ND1 53325212 IC50 > 150000 nM T85943 CR0U8Q 53326498 IC50 = 108700 nM T85943 CX4M7F 53326500 IC50 = 105500 nM T85943 C1Y7CJ 53326745 IC50 = 12700 nM T85943 C1KYR9 53326941 IC50 > 50000 nM T85943 C5EOS8 53328013 IC50 = 520 nM T85943 CVC5T4 53328120 IC50 = 5900 nM T85943 C9PR3G 53328121 IC50 = 1300 nM T85943 C8WJC1 53328317 IC50 = 4500 nM T85943 C4R1OF 53328318 IC50 = 96000 nM T85943 C2YC0W 53328319 IC50 = 3600 nM T85943 CJIE57 53328320 IC50 = 22000 nM T85943 C6XQ3O 53328321 IC50 = 40000 nM T85943 CKQA18 53328322 IC50 = 1900 nM T85943 CHC90P 53328509 IC50 = 620 nM T85943 CNG20E 53328510 IC50 = 720 nM T85943 CA2N6W 53328511 IC50 = 380 nM T85943 C72RMJ 53328512 IC50 = 2800 nM T85943 CB64PJ 53344791 IC50 > 10000 nM T85943 C34WUD 53344792 IC50 = 3100 nM T85943 CKMT06 53344794 IC50 > 10000 nM T85943 CX09YO 53344795 IC50 = 1800 nM T85943 C8B4YV 53344796 IC50 = 380 nM T85943 COA40N 53344910 IC50 = 41 nM T85943 CTPD39 53344911 IC50 = 200 nM T85943 CT36PS 53344912 IC50 = 780 nM T85943 C35KDN 53344913 IC50 = 260 nM T85943 CS2F7B 53344914 IC50 > 10000 nM T85943 C76HBP 53344915 IC50 = 280 nM T85943 C5EVU4 53345021 IC50 = 280 nM T85943 CJ6GR7 53345135 IC50 = 270 nM T85943 CFG8M4 53346428 IC50 = 550 nM T85943 C38IEN 53346429 IC50 = 300 nM T85943 C9D0TP 53346431 Ki > 20000 nM T85943 COA86E 53346433 IC50 > 10000 nM T85943 C0SWH5 53348216 IC50 > 40000 nM T85943 C8ZRE3 53356518 IC50 = 2434 nM T85943 CM7P3W 53357328 IC50 = 250 nM T85943 CBK9Q6 53357848 IC50 > 10000 nM T85943 CJ7R1T 53358198 IC50 = 50600 nM T85943 CR7KQ9 53358307 IC50 = 58300 nM T85943 CHF3Q9 53358308 IC50 = 98300 nM T85943 CPR62M 53358309 IC50 = 60500 nM T85943 CSUD43 53358310 IC50 = 87000 nM T85943 CY2W7C 53358311 IC50 > 150000 nM T85943 CX6NY0 53358312 IC50 > 150000 nM T85943 CV7KR8 53358313 IC50 = 106000 nM T85943 C8NA4L 53384644 IC50 > 30000 nM T85943 CBS73R 53484203 Ki = 90 nM T85943 CUWH19 54580280 IC50 = 63 nM T85943 C6QV2U 54580281 IC50 = 3870 nM T85943 C1NR6H 54581279 IC50 = 330 nM T85943 C0M4OX 54581587 IC50 > 150000 nM T85943 CHZL12 54581588 IC50 = 100000 nM T85943 CG1PJ5 54582301 IC50 = 2080 nM T85943 CU0YE9 54582578 IC50 > 150000 nM T85943 C3NL6S 54582579 IC50 > 150000 nM T85943 COQ42Z 54583273 IC50 = 769 nM T85943 CF4VM8 54583274 IC50 = 1300 nM T85943 CYB91O 54583275 IC50 = 107 nM T85943 CI7FT4 54583276 IC50 = 68 nM T85943 CPF70C 54583551 IC50 > 150000 nM T85943 C7PJZ9 54584237 IC50 = 230 nM T85943 CIO84P 54584531 IC50 = 71600 nM T85943 CH01MG 54585208 IC50 > 10000 nM T85943 C0XLS5 54585209 IC50 = 840 nM T85943 CANJ42 54585467 IC50 > 150000 nM T85943 C3YA2X 54585879 Ki = 7140 nM T85943 CNH30M 54586160 IC50 = 1340 nM T85943 CT3B8X 54586437 IC50 > 150000 nM T85943 CHX1Y5 54587168 IC50 > 10000 nM T85943 C7CF2E 54587466 IC50 > 150000 nM T85943 C1XS2J 54760383 IC50 = 290 nM T85943 C9ZFS1 54764923 IC50 = 2400 nM T85943 CM8JX1 56604907 IC50 = 10 nM T85943 CUSJ18 56657888 IC50 = 80700 nM T85943 CM4BL9 56657889 IC50 = 69500 nM T85943 C8X5VW 56658814 IC50 < 500 nM T85943 C3IGE9 56661327 IC50 = 12100 nM T85943 C6DYM0 56661328 IC50 > 100000 nM T85943 CJV63Y 56662161 Ki = 480 nM T85943 CA51VH 56662318 Ki = 2160 nM T85943 C1MUS9 56662319 Ki = 2810 nM T85943 C3B6TD 56662320 Ki = 2000 nM T85943 CJV01G 56664629 IC50 > 700000 nM T85943 C9M6CD 56664866 IC50 = 75400 nM T85943 CAR67O 56665753 Ki = 25 nM T85943 C29HIE 56668275 IC50 = 1500 nM T85943 CLXT42 56671742 IC50 > 100000 nM T85943 C9F0OE 56674968 IC50 = 17000 nM T85943 CAFS10 56675105 IC50 = 90700 nM T85943 CG57QJ 56675166 IC50 = 1100 nM T85943 CI8E5L 56675167 IC50 = 5900 nM T85943 C8HSU5 56675168 IC50 = 1200 nM T85943 CLHO15 56676037 Ki = 25 nM T85943 CE0B2Y 56678464 IC50 = 3300 nM T85943 C0QFK5 56679360 Ki = 510 nM T85943 CD3GF9 56681625 IC50 = 400000 nM T85943 CI2T5P 56681756 IC50 > 100000 nM T85943 CQ5Z1I 56681809 IC50 > 100000 nM T85943 C0UI3E 56682663 Ki = 18 nM T85943 CBOD63 56835089 IC50 > 30000 nM T85943 CIK1P3 56835114 IC50 = 35100 nM T85943 CC06BM 56835765 Ki > 10000 nM T85943 CLNY43 56835766 Ki > 10000 nM T85943 CCR71V 56835771 Ki > 10000 nM T85943 C9CJ7B 56835772 IC50 > 10000 nM T85943 C5SW6Q 56930741 IC50 = 86000 nM T85943 CR16SD 56947170 IC50 = 840 nM T85943 CGQ94I 56950740 IC50 = 6400 nM T85943 CN1XL0 56950741 IC50 > 100000 nM T85943 C3ER0V 56950742 IC50 = 19000 nM T85943 CEZ14X 56950743 IC50 = 55000 nM T85943 CTL49B 56950878 IC50 > 100000 nM T85943 CM5HO1 56950881 IC50 = 52000 nM T85943 C9CLJ0 56950882 IC50 = 23000 nM T85943 CG0VC7 56950883 IC50 = 23000 nM T85943 CE1GO5 56950884 IC50 = 82000 nM T85943 CLQ4Z9 56950885 IC50 = 53000 nM T85943 C40BPN 56951005 IC50 > 100000 nM T85943 CL9XP2 56951006 IC50 = 6700 nM T85943 CKV5O2 56951007 IC50 = 2000 nM T85943 C97QIR 56951008 IC50 = 12000 nM T85943 CP58NG 56954518 IC50 = 5470 nM T85943 CAK91L 56955954 IC50 > 3600 nM T85943 CT8ZB0 56963800 IC50 = 2000 nM T85943 CJ47MX 56963907 IC50 = 5600 nM T85943 C9L6FD 56963908 IC50 > 10000 nM T85943 CE50IB 56963909 IC50 > 10000 nM T85943 CPHX64 57325478 IC50 > 50000 nM T85943 CQ9BW4 57325479 IC50 > 50000 nM T85943 CF6K7P 57391515 IC50 > 150000 nM T85943 C03CTS 57391516 IC50 = 82700 nM T85943 CSMQ30 57391517 IC50 = 58400 nM T85943 CNS23O 57393341 IC50 > 150000 nM T85943 C1LD7K 57393342 IC50 = 66600 nM T85943 CE1A9V 57394653 IC50 = 84 nM T85943 CNV76Z 57394656 IC50 = 410 nM T85943 CEN37G 57394999 IC50 = 57700 nM T85943 CZ2B4I 57395000 IC50 > 150000 nM T85943 CD6Y9Z 57395116 IC50 > 30000 nM T85943 C8W6IG 57395117 IC50 > 30000 nM T85943 CJKC17 57395223 IC50 = 81000 nM T85943 C3KQY5 57396743 IC50 > 150000 nM T85943 C1AY8Q 57396744 IC50 = 74300 nM T85943 CPID34 57396826 IC50 > 150000 nM T85943 CBFC15 57396827 IC50 = 50700 nM T85943 CG7S0D 57396882 IC50 > 30000 nM T85943 C8JXE3 57398517 IC50 > 150000 nM T85943 C6KO5E 57398518 IC50 > 150000 nM T85943 CKV7A8 57398519 IC50 > 150000 nM T85943 CT7QD5 57400187 IC50 > 150000 nM T85943 C4OY0K 57400188 IC50 > 150000 nM T85943 CV7PL9 57400250 IC50 > 150000 nM T85943 CC0BD6 57400251 IC50 > 150000 nM T85943 C1O8JK 57401981 IC50 = 131800 nM T85943 C45EAQ 57401982 IC50 > 150000 nM T85943 CAJ0E6 57402051 IC50 = 94100 nM T85943 CWX45G 57402052 IC50 = 62100 nM T85943 CA5P0J 57402053 IC50 > 150000 nM T85943 CD03QW 57402054 IC50 > 150000 nM T85943 CYL5E6 57403737 IC50 > 150000 nM T85943 CBR0U6 57403738 IC50 = 77300 nM T85943 CQ9R7G 57403800 IC50 > 150000 nM T85943 CP5QO9 57403801 IC50 > 150000 nM T85943 C0GAM8 57403802 IC50 > 150000 nM T85943 C53WAD 57403803 IC50 = 65800 nM T85943 CVK0G4 58056356 IC50 > 50000 nM T85943 CPOF74 58159418 IC50 = 483900 nM T85943 CWXC70 58180596 IC50 > 2000 nM T85943 C3VI7D 58229394 IC50 = 995 nM T85943 CNXU29 58229412 IC50 = 113 nM T85943 C52OMW 58229434 IC50 = 1723 nM T85943 CV13QY 58540422 IC50 = 924 nM T85943 CQJX07 59073929 IC50 = 320 nM T85943 CZ2RN3 59073937 IC50 = 400 nM T85943 CXJ63M 59603829 IC50 = 42 nM T85943 CQEU96 59603842 IC50 = 3 nM T85943 CP89BI 59633491 IC50 > 10000 nM T85943 CX8Y0E 59633494 IC50 = 607 nM T85943 CKE14A 59633616 IC50 > 10000 nM T85943 C0QUY4 59633665 IC50 > 10000 nM T85943 CT62RM 59633704 IC50 > 10000 nM T85943 CBPQ52 59633728 IC50 > 10000 nM T85943 C0QRM9 59633812 IC50 > 10000 nM T85943 CLH49Z 59790029 IC50 = 2 nM T85943 COH62U 60097413 IC50 > 3300 nM T85943 C1MR8Q 60097495 IC50 > 5000 nM T85943 CSZA16 60155724 IC50 > 3600 nM T85943 CU79HD 60202383 IC50 = 32 nM T85943 C9ZCT2 62705065 IC50 > 1000 nM T85943 CUBL90 66545750 IC50 = 338 nM T85943 CK6WO0 66552478 IC50 < 10000 nM T85943 CDE5J0 66552525 IC50 > 10000 nM T85943 CI3J2H 66552648 IC50 > 10000 nM T85943 CA9Z7N 66552722 IC50 > 10000 nM T85943 CT6D3Y 66552723 IC50 > 10000 nM T85943 C2DL4Q 66552781 IC50 > 10000 nM T85943 CXB5R0 66552850 IC50 > 10000 nM T85943 C9O4GF 66555232 IC50 = 16000 nM T85943 CL3EN2 66556938 IC50 > 50000 nM T85943 C9QF6B 66559005 IC50 = 645 nM T85943 CD14OC 67071561 IC50 = 1951 nM T85943 CEKN37 67073846 IC50 = 44 nM T85943 CE49GC 67098566 Ki = 480 nM T85943 CV63UL 67240318 IC50 > 10000 nM T85943 CO6W9D 68004741 IC50 = 300 nM T85943 CB6U7F 68005465 IC50 = 510 nM T85943 CK83VI 68005486 IC50 > 50000 nM T85943 C1RJ7Y 68005600 IC50 = 7000 nM T85943 COX3U9 68005621 IC50 = 390 nM T85943 CEXN58 68005732 IC50 = 2000 nM T85943 CWF1M9 68263732 Ki > 20000 nM T85943 C8I7GC 68293638 IC50 > 10000 nM T85943 CAIO65 68796885 IC50 = 40 nM T85943 CHMB14 68925961 IC50 = 1000 nM T85943 C5DGR9 69036886 IC50 = 668 nM T85943 CCU8A1 69912574 IC50 = 184700 nM T85943 C7VJ6A 70647728 IC50 = 3190 nM T85943 C7YCR9 70681746 IC50 = 41.2 nM T85943 C81LEG 70681747 IC50 = 385 nM T85943 C3QMI8 70682505 IC50 > 10000 nM T85943 CVQP45 70682511 IC50 > 10000 nM T85943 C6C5GY 70682512 IC50 > 10000 nM T85943 C4NM9V 70682513 Ki > 10000 nM T85943 CLB70A 70682515 IC50 = 4100 nM T85943 CSM23I 70682523 IC50 > 10000 nM T85943 CU10OI 70682525 IC50 = 6700 nM T85943 CW80GP 70683852 IC50 = 155 nM T85943 C5W3UA 70683853 IC50 = 188 nM T85943 CRI43A 70684578 IC50 > 10000 nM T85943 C60JBH 70684595 IC50 > 10000 nM T85943 C4XN7E 70684597 IC50 = 1600 nM T85943 C6PK1Z 70684599 IC50 > 10000 nM T85943 CI7ZK3 70685991 IC50 = 25.1 nM T85943 CO7X6N 70685992 IC50 = 43.1 nM T85943 CM6B2X 70686729 IC50 = 130 nM T85943 CTO8Y7 70686730 IC50 = 1300 nM T85943 C2FR0M 70686734 IC50 = 2100 nM T85943 CDGH36 70686735 IC50 = 2200 nM T85943 C1P5LT 70686736 IC50 > 10000 nM T85943 C83LEN 70686737 IC50 = 65 nM T85943 C9M1UN 70686738 IC50 = 200 nM T85943 CE2YM0 70686739 IC50 > 10000 nM T85943 C5E1ZL 70686750 IC50 > 10000 nM T85943 C82FIP 70686752 IC50 = 380 nM T85943 C34WBD 70686758 IC50 = 8700 nM T85943 CE1DK6 70686760 IC50 = 3300 nM T85943 C45EPC 70686762 IC50 = 5200 nM T85943 C0QX3Y 70688829 IC50 = 670 nM T85943 C29IWN 70688831 IC50 = 2200 nM T85943 C7MA3L 70688835 IC50 > 10000 nM T85943 C1OLS7 70690770 IC50 = 3100 nM T85943 C08VID 70690904 IC50 > 10000 nM T85943 CDUS20 70690906 IC50 = 5100 nM T85943 CEM0Q4 70690908 IC50 = 520 nM T85943 C5C0KE 70690925 IC50 = 1600 nM T85943 CUS3F6 70691280 IC50 = 1900 nM T85943 C8D3MF 70692306 IC50 = 8.8 nM T85943 CBS26Q 70692909 IC50 = 7500 nM T85943 C17AVH 70693049 IC50 = 120 nM T85943 CSOT12 70693058 IC50 > 10000 nM T85943 CS6NW3 70693059 IC50 > 10000 nM T85943 C05LUE 70693064 IC50 > 10000 nM T85943 CJW6U8 70694945 IC50 = 66000 nM T85943 CA76MR 70695090 IC50 = 650 nM T85943 CW8RU1 70695091 IC50 = 8800 nM T85943 CX73CN 70695104 IC50 = 5000 nM T85943 C2JHC8 70695106 IC50 = 730 nM T85943 CBT3M4 70695108 IC50 = 810 nM T85943 CH8N1I 70695110 IC50 = 8200 nM T85943 CHC4I6 70695497 IC50 = 2600 nM T85943 C8LV5X 70697131 IC50 = 180 nM T85943 CA9R3F 70697140 IC50 = 1100 nM T85943 C4YBV3 70697145 IC50 > 10000 nM T85943 CRH9B4 70697147 IC50 > 10000 nM T85943 C1EBC8 70697149 IC50 = 6300 nM T85943 CCAR97 70697516 IC50 = 2800 nM T85943 CK1B7F 70697575 IC50 = 403 nM T85943 C1IEJ2 70789254 IC50 = 150000 nM T85943 C8T7ZP 70789255 IC50 = 18000 nM T85943 CH0B8N 70789756 IC50 > 30000 nM T85943 CK2QM6 70866006 IC50 = 3037 nM T85943 CV74OC 70866036 IC50 = 1167 nM T85943 CMX75Z 70866164 IC50 = 54 nM T85943 CVNH21 70866177 IC50 = 209 nM T85943 CKJI02 70866181 IC50 = 1473 nM T85943 COU73Y 71226944 IC50 = 55 nM T85943 C40JOZ 71235465 IC50 = 123 nM T85943 C91HPI 71300299 IC50 > 5000 nM T85943 C8DR6V 71450494 IC50 = 297300 nM T85943 CX7AB0 71450495 IC50 = 125000 nM T85943 C8BEJ7 71450496 IC50 = 451000 nM T85943 CEBO91 71452977 IC50 > 10000 nM T85943 C2S1PA 71454126 IC50 = 224800 nM T85943 CKT60L 71455860 Ki > 1900 nM T85943 C1F8BT 71457659 IC50 = 143400 nM T85943 CAR8F7 71457660 IC50 = 95000 nM T85943 C9DIK2 71512060 IC50 = 1731 nM T85943 C5ZKU7 71546969 IC50 = 71 nM T85943 C7ARI9 71547113 IC50 = 110 nM T85943 CA3O6K 71552696 IC50 = 3690 nM T85943 C1NPL0 71552941 IC50 > 30000 nM T85943 CA4PS8 71552942 IC50 > 30000 nM T85943 CB3SO2 71567006 IC50 > 10000 nM T85943 CDJY72 71568837 IC50 > 10000 nM T85943 CN7W5S 71579325 IC50 > 10000 nM T85943 C6VNW7 71624837 IC50 = 25000 nM T85943 CYL9T4 71625080 IC50 = 46900 nM T85943 CQ17MK 71625214 IC50 = 7100 nM T85943 C7X8UK 71625332 IC50 = 69100 nM T85943 C7E6YV 71720026 IC50 = 46 nM T85943 CI4N7R 71745294 Ki = 165 nM T85943 CRC14G 71745295 Ki = 1700 nM T85943 CCQE91 71745296 Ki = 1097 nM T85943 C5Z8IT 71745297 Ki = 723 nM T85943 C9D5PT 71745298 Ki = 770 nM T85943 CAJ13X 71745299 Ki = 150 nM T85943 CN91IU 71745494 Ki = 637 nM T85943 C7SUW0 71747648 Ki = 45 nM T85943 CE5KF3 71747828 Ki = 1400 nM T85943 C7HJG1 71747829 Ki = 340 nM T85943 CRU82Q 71747830 Ki = 395 nM T85943 CGKP21 71747831 Ki = 2350 nM T85943 CAQ1W4 71747832 Ki = 110 nM T85943 CE3A9T 71747833 Ki = 60 nM T85943 C4GJ1V 71747834 Ki = 618 nM T85943 C14EQL 71748013 Ki = 70 nM T85943 COZT25 71748014 Ki = 620 nM T85943 C6BN2O 71748015 Ki = 6 nM T85943 CHWO28 71748016 Ki = 610 nM T85943 CUQW27 71748017 Ki = 500 nM T85943 CM82AO 71748018 Ki = 1080 nM T85943 CS4E9X 71762922 Ki > 100000 nM T85943 CZM1K4 71765510 IC50 = 67 nM T85943 CPV93K 71814883 IC50 = 14500 nM T85943 CR94ZB 72164776 Ki = 371 nM T85943 CI9H6L 72164895 Ki = 138 nM T85943 CF17AG 72164896 Ki = 190 nM T85943 CGPN68 72164897 Ki = 407 nM T85943 C6HG5M 72164898 Ki = 4300 nM T85943 C7W0GL 72164899 Ki = 2140 nM T85943 C64BDO 72165040 Ki > 12500000 nM T85943 CV12UF 72736749 IC50 = 27.3 nM T85943 C62TJC 73254853 IC50 > 30000 nM T85943 C0HSC8 73346520 Ki = 15310 nM T85943 C8SD9P 73346521 Ki = 20170 nM T85943 CGZ6Y8 73346522 Ki = 16690 nM T85943 CE1MQ2 73347352 IC50 >= 300000 nM T85943 CIN46S 73347353 IC50 = 21500 nM T85943 C43IPQ 73348006 Ki = 3230 nM T85943 C60PDQ 73350151 IC50 = 5000 nM T85943 C4L7IR 73350439 IC50 = 52600 nM T85943 CU5YN3 73350440 IC50 = 31300 nM T85943 CS9C0W 73351108 Ki = 4730 nM T85943 C27JUH 73352576 Ki = 14760 nM T85943 CVP03Z 73352577 Ki = 7910 nM T85943 CX75YR 73352604 IC50 = 39.81 nM T85943 CDAB86 73354065 Ki = 13480 nM T85943 CK3Z8U 73354066 Ki = 14130 nM T85943 C92DXZ 73354067 Ki = 13270 nM T85943 CCI18Y 73355591 Ki = 1900 nM T85943 CRX8A0 73355592 Ki = 34300 nM T85943 CSUZ81 73356106 IC50 = 160000 nM T85943 C60IFK 73356254 IC50 = 16000 nM T85943 CY40RW 73356484 IC50 = 1567600 nM T85943 C2UC1B 73356485 IC50 >= 300000 nM T85943 C90UXA 73356487 IC50 >= 300000 nM T85943 C6UA4K 73356522 IC50 > 3000 nM T85943 CZ0C5Y 73670809 IC50 = 1320 nM T85943 CM3Y6X 73670970 IC50 = 7270 nM T85943 CC3AG1 73670971 IC50 = 980 nM T85943 CR85PZ 73670972 IC50 = 2700 nM T85943 CB8DI0 73670973 IC50 = 6930 nM T85943 CV8KI3 73670975 IC50 > 10000 nM T85943 CX1LR9 73774633 IC50 = 4030 nM T85943 C3UC9H 73891099 IC50 = 370 nM T85943 CS9BQ1 74222426 IC50 = 1400 nM T85943 CO0V6K 74222427 IC50 = 1630 nM T85943 CBE71O 74222509 IC50 > 20000 nM T85943 CM02PA 74222510 IC50 = 4.2 nM T85943 CWLT81 74222511 IC50 = 14400 nM T85943 C4XSG8 74222512 IC50 = 5840 nM T85943 CBT4M6 74222513 IC50 = 3140 nM T85943 C53AFH 74222599 IC50 = 4610 nM T85943 C8W2HV 76309526 Ki < 100 nM T85943 CV8QX0 76310169 IC50 = 12600 nM T85943 C6D0LO 76316736 Ki < 100 nM T85943 CA5L4W 76324771 IC50 = 20000 nM T85943 C9GO0P 76328313 IC50 = 3560 nM T85943 CJ2T9E 76332983 IC50 = 3040 nM T85943 C39FTZ 76335685 IC50 = 19700 nM T85943 CH8W7D 77461036 IC50 > 1000 nM T85943 CWG4T2 78209992 IC50 = 622 nM T85943 CSH3G2 86287525 IC50 > 60000 nM T85943 CB5NJ4 86302541 IC50 > 10000 nM T85943 CPG3A5 86302574 IC50 = 15453 nM T85943 C5ZI4L 86341927 IC50 = 4750 nM T85943 CH62SW 86341928 IC50 > 10000 nM T85943 CTJ2H7 86341929 IC50 > 10000 nM T85943 CFZB81 86341930 IC50 > 10000 nM T85943 CDAY96 86341931 IC50 > 10000 nM T85943 CB3RM9 86341934 IC50 > 10000 nM T85943 CC32NJ 86342041 IC50 > 10000 nM T85943 CSQO18 86342043 IC50 > 10000 nM T85943 CZI4Q8 86342076 IC50 > 10000 nM T85943 C5T2GX 86342077 IC50 > 10000 nM T85943 C2T9BN 86342078 IC50 > 10000 nM T85943 C4EQ8X 86342079 IC50 > 10000 nM T85943 C6XJF9 86342081 IC50 > 10000 nM T85943 C4VL7Y 86342082 IC50 > 30000 nM T85943 CMK19R 86342113 IC50 > 30000 nM T85943 C73LNE 86342141 IC50 > 10000 nM T85943 CCP67Y 86342144 IC50 > 10000 nM T85943 C7CL5Y 86342146 IC50 > 10000 nM T85943 CTX6G7 86342496 IC50 > 10000 nM T85943 C0AN7G 86342862 IC50 > 10000 nM T85943 CH32AN 86343050 IC50 = 10000 nM T85943 CH7U9K 86343056 IC50 = 3300 nM T85943 C1HW4B 89735655 IC50 = 8100 nM T85943 C0AK9G 89891791 IC50 = 1127 nM T85943 CT7KE8 89891806 IC50 = 29 nM T85943 C73PSN 89891847 IC50 = 51 nM T85943 CBW32H 89899386 IC50 = 168 nM T85943 CTY2A0 89899410 IC50 = 759 nM T85943 CPVZ54 89899415 IC50 = 9.5 nM T85943 CJYP54 89899416 IC50 = 2224 nM T85943 CSM02W 89899417 IC50 = 3.4 nM T85943 CDAU89 89899421 IC50 = 12 nM T85943 CR3XL7 90119070 IC50 = 3350 nM T85943 CLK3O0 90119255 IC50 = 6480 nM T85943 CO2FV0 90119264 IC50 = 72 nM T85943 C3RL4C 90136268 IC50 = 3410 nM T85943 C4ME0V 90136282 IC50 > 20000 nM T85943 CY0T6O 90136348 IC50 = 370 nM T85943 CFB75T 90479825 IC50 = 438 nM T85943 C3GU7P 90645237 IC50 > 10000 nM T85943 CFI93O 90645239 IC50 > 10000 nM T85943 C76KSB 90645241 IC50 > 10000 nM T85943 CNWP80 90645243 IC50 > 10000 nM T85943 C1POJ2 90645244 IC50 > 10000 nM T85943 C8BEX4 90645245 IC50 > 10000 nM T85943 CCWY46 90657091 Ki = 200 nM T85943 C14YHF 90663234 IC50 = 350 nM T85943 CO5I7X 90663263 IC50 = 5000 nM T85943 CUIW21 90663264 IC50 = 5500 nM T85943 CR1W4U 90663267 IC50 = 4500 nM T85943 C09HAT 90663283 IC50 = 3400 nM T85943 CN2R9H 90663284 IC50 = 20000 nM T85943 CZ23BX 90663285 IC50 = 1400 nM T85943 C24QVG 91933026 IC50 = 17000 nM T85943 C9TD4S 91933027 IC50 = 20000 nM T85943 C0Y8ZK 91933875 IC50 > 100 nM T85943 CJQ5N6 91936970 IC50 = 1010000 nM T85943 CB8AR9 91970527 IC50 = 254 nM T85943 CCVL49 100942265 IC50 = 81000 nM T85943 C24SBM 101338350 IC50 = 1600 nM T85943 C41DFX 101913643 Ki = 130 nM T85943 CJIA82 117704411 IC50 > 10000 nM T85943 C9MJE1 118226293 Ki = 0.261 nM T85943 C3KLI5 118723185 IC50 > 100000 nM T85943 CLV8J2 118725186 IC50 = 52 nM T85943 CU09DP 118725208 IC50 = 2300 nM T85943 CY8MG4 118725828 Ki = 230 nM T85943 C1DSM9 118725829 Ki = 1460 nM T85943 C39WRI 118725830 Ki = 1060 nM T85943 CY58OQ 118725831 Ki = 200 nM T85943 CVT97W 118725832 Ki = 620 nM T85943 CW2JN4 118725833 Ki = 1200 nM T85943 C4DU6M 118725835 Ki = 40 nM T85943 C92XHV 118725866 Ki = 790 nM T85943 C2X4TB 118725867 Ki = 550 nM T85943 CAHN07 118725868 Ki = 100 nM T85943 CWJ7B5 118725869 Ki = 110 nM T85943 CUI1O8 118725870 Ki = 1440 nM T85943 CESR14 118725871 Ki = 2340 nM T85943 CKT21A 118725872 Ki = 970 nM T85943 CA9GJ0 118725874 Ki = 70 nM T85943 CJST86 118725875 Ki = 30 nM T85943 C71XZR 118725876 Ki = 130 nM T85943 C0FEJ7 118725877 Ki = 300 nM T85943 C61DWI 118725878 Ki = 260 nM T85943 C6U1WL 118725879 Ki = 620 nM T85943 C25DKS 118725880 Ki = 10 nM T85943 CH9N4T 118725881 Ki = 120 nM T85943 CLEW12 118725882 Ki = 110 nM T85943 CO4CN9 118725884 Ki = 7 nM T85943 CHT6K9 118728811 Ki > 4000 nM T85943 CUA3Y2 118728812 Ki > 4000 nM T85943 CDQ78G 118728813 Ki > 4000 nM T85943 CZ6XL7 118728814 Ki > 4000 nM T85943 CMO67K 118728815 Ki > 4000 nM T85943 CR2M0Q 118728816 Ki > 4000 nM T85943 C62SCL 118728817 Ki > 4000 nM T85943 CSB30C 118728819 Ki = 3100 nM T85943 CV7XU8 118728820 Ki = 3500 nM T85943 C3J1EX 118728821 Ki > 4000 nM T85943 CIWB78 118728822 Ki = 2500 nM T85943 CP18SE 118728823 Ki = 970 nM T85943 CM42CA 118728824 Ki = 2400 nM T85943 C9Q7CL 118728825 Ki > 4000 nM T85943 CCR3S0 118728826 Ki = 3100 nM T85943 CIT9X6 118737048 IC50 = 2 nM T85943 CW0X7N 118737049 IC50 = 4 nM T85943 CLFM69 118737050 IC50 = 2 nM T85943 C8R5QJ 118737051 IC50 = 1 nM T85943 C21FCW 118737052 IC50 = 3 nM T85943 C3V9KL 118737053 IC50 = 21 nM T85943 C2CF1W 118737054 IC50 = 2 nM T85943 CFW54Z 118737055 IC50 = 4 nM T85943 CUN41S 118737056 IC50 = 7 nM T85943 CQCX41 118737057 IC50 = 0.9 nM T85943 C93GZM 118737058 IC50 = 9 nM T85943 C2R3XA 118737059 IC50 = 19 nM T85943 C7PSY9 118737060 IC50 = 8 nM T85943 CYR36N 118737061 IC50 = 7 nM T85943 CG2K3O 118737062 IC50 = 7 nM T85943 CO1QM3 118737064 IC50 = 12 nM T85943 C1POS5 118737065 IC50 = 15 nM T85943 C3E4OP 118737066 IC50 = 5 nM T85943 CAB57R 118737067 IC50 = 11 nM T85943 CU81ZN 118737068 IC50 = 83 nM T85943 C9UHW7 118737069 IC50 = 1409 nM T85943 COW3Y0 118737071 IC50 = 59 nM T85943 C05AOM 118737072 IC50 = 3191 nM T85943 CKBP72 121231408 IC50 < 0.5 nM T85943 CP0S5T 121246673 IC50 > 10000 nM T85943 C1Y7UH 121305843 Ki > 100000 nM T85943 CHG8Y6 121316022 Ki > 100000 nM T85943 C81IFQ 122163152 IC50 > 100000 nM T85943 C08KEM 122179540 IC50 = 4600 nM T85943 CG0RP7 122179547 IC50 = 2500 nM T85943 C1A0SQ 122179548 IC50 = 4600 nM T85943 C42GSX 122180520 Ki > 4000 nM T85943 CM5FZ6 122186141 IC50 = 28 nM T85943 CA3SU2 122186150 IC50 = 17 nM T85943 CI8RS6 122186151 IC50 = 260 nM T85943 CK70HC 122188437 IC50 = 36500 nM T85943 C9XA3B 122188439 IC50 = 21600 nM T85943 C2E8ID 122188441 IC50 = 73500 nM T85943 C10QOD 122190497 Ki = 360 nM T85943 C8HF2J 122190498 Ki = 200 nM T85943 CCXA46 122190499 Ki = 400 nM T85943 CC0MD7 122190500 Ki = 90 nM T85943 CJT7M3 122190501 Ki = 140 nM T85943 C4ZU8S 122190502 Ki = 480 nM T85943 CD6B0A 122190503 Ki = 230 nM T85943 CRC82U 122190504 Ki = 330 nM T85943 C3PQ4W 122190505 Ki = 70 nM T85943 CY8P9C 122190506 Ki = 370 nM T85943 CN1DK0 122190507 Ki = 130 nM T85943 CNX0Q2 122193763 IC50 > 10000 nM T85943 CWV0C3 122193764 IC50 > 10000 nM T85943 CSG98Y 122193765 IC50 = 7640 nM T85943 CCLQ75 122193769 IC50 > 10000 nM T85943 CXDR48 122193770 IC50 > 10000 nM T85943 CPA8C5 122193773 IC50 = 8460 nM T85943 CN41IF 122634050 IC50 = 90 nM T85943 CD67LU 122705248 IC50 = 27 nM T85943 CX63VW 122705258 IC50 = 1040 nM T85943 C76IKM 122705261 IC50 = 2450 nM T85943 CY30FL 123752658 IC50 = 10.8 nM T85943 C8ALO2 124088839 IC50 = 303 nM T85943 CK46IZ 124088840 IC50 = 3.5 nM T85943 CKC81N 124088842 IC50 = 194 nM T85943 C2XIS6 124088843 IC50 = 71 nM T85943 CXVU91 124088862 IC50 = 114 nM T85943 COBA69 124088864 IC50 = 1 nM T85943 CBLA08 124088870 IC50 = 0.6 nM T85943 CX3O4K 124088871 IC50 > 10000 nM T85943 C4OH5B 124088876 IC50 = 1 nM T85943 C8KXV1 127025843 IC50 > 1000 nM T85943 CKS28E 127034802 IC50 = 75.4 nM T85943 CKX40V 127037812 IC50 > 10000 nM T85943 C70RUP 127038480 IC50 > 10000 nM T85943 C3WCN8 127041777 IC50 > 10000 nM T85943 CG8DA9 127045861 IC50 > 100000 nM T85943 CHK16Q 127045929 IC50 > 1000 nM T85943 CC4ND8 127046862 IC50 > 100000 nM T85943 CY3J0C 127047591 IC50 > 1000 nM T85943 COPL97 127049453 IC50 < 0.5 nM T85943 CDP32G 127050839 IC50 = 21 nM T85943 CO25WH 127052538 IC50 = 126 nM T85943 CA5XE4 129012139 IC50 > 10000 nM T85943 CKJT41 129316172 IC50 > 10000 nM T85943 CHC0A7 129900194 IC50 = 828 nM T85943 C8F0DQ 129909860 IC50 = 93 nM T85943 C0FM1R 130196825 IC50 = 1053 nM T85943 C43ECX 130431658 IC50 > 10000 nM T85943 CO45HN 130431659 IC50 > 10000 nM T85943 CH2S1Y 130431660 IC50 > 10000 nM T85943 CN5EI1 130431665 IC50 > 10000 nM T85943 C3BK5P 130431668 IC50 > 10000 nM T85943 CYI5W6 130431670 IC50 > 10000 nM T85943 C73XET 130431673 IC50 > 10000 nM T85943 CJ6I3R 130431677 IC50 > 10000 nM T85943 C9Q1AR 130431683 IC50 > 10000 nM T85943 C64JHD 130431688 IC50 > 10000 nM T85943 C05GIE 130431689 IC50 > 10000 nM T85943 C69TKF 130431691 IC50 > 10000 nM T85943 C7GMX3 130431694 IC50 > 10000 nM T85943 CNE46K 130431700 IC50 > 10000 nM T85943 C1AG2J 130431702 IC50 = 901 nM T85943 CH09QX 130431745 IC50 > 10000 nM T85943 C8FW7S 130434411 IC50 > 10000 nM T85943 C8ARK0 131801160 IC50 = 4 nM T85943 CERS64 132937256 IC50 > 30000 nM T85943 C98MZB 134132731 IC50 = 4700 nM T85943 C6B1EN 134133066 IC50 = 3330 nM T85943 CZG2L5 134135232 IC50 = 24000 nM T85943 CK9W4F 134135741 IC50 = 250 nM T85943 C7SL4N 134143939 IC50 = 67000 nM T85943 CMA60G 134144799 IC50 = 33000 nM T85943 C3MN6B 134144868 IC50 = 11 nM T85943 CEZH84 134146580 IC50 = 230 nM T85943 CN35SO 134146628 IC50 > 1000 nM T85943 C1DF4R 134147544 IC50 = 31 nM T85943 C95NCV 134151662 IC50 = 0.18 nM T85943 CX7YE1 134155961 IC50 = 330 nM T85943 CE38MW 134156584 IC50 = 0.43 nM T85943 CVI25K 134157526 IC50 = 4.3 nM T85943 C2AN7T 134611886 IC50 > 100000 nM T85943 CYL5V1 134694986 IC50 = 17056 nM T85943 C6X4LW 134816069 Ki = 18 nM T85943 CK7RY6 134816070 Ki = 22 nM T85943 CSZM60 134816433 Ki = 200 nM T85943 CNK2R8 134816533 Ki = 710 nM T85943 CJ2XB5 135398585 IC50 > 100000 nM T85943 CVJK60 135402835 IC50 = 8550 nM T85943 CJ1I5M 135402981 IC50 = 75 nM T85943 CH97JB 135402982 IC50 = 16 nM T85943 C26GSU 135402983 IC50 = 30 nM T85943 CK8EJ6 135402984 IC50 = 330 nM T85943 CHS5X0 135409466 IC50 = 0.2 ug.mL-1 T85943 C2DH1R 135412832 IC50 = 0.225 ug.mL-1 T85943 CO7DF9 135423833 IC50 = 200 nM T85943 C2B6JR 135436036 IC50 = 293000 nM T85943 C50VLW 135443391 IC50 = 41000 nM T85943 C8GZ2B 135449326 Ki = 1100 nM T85943 C19YWA 135457035 Ki = 500 nM T85943 C8NTH5 135503520 IC50 = 35 nM T85943 CU97NR 135510708 IC50 = 430 nM T85943 C08KLE 135520206 IC50 = 13 nM T85943 CLK9D1 135523696 IC50 = 500 nM T85943 CTB7R2 135564980 IC50 = 250 nM T85943 CY4D8I 135566504 Ki > 1000 nM T85943 CRJ45X 135589980 IC50 > 50000 nM T85943 CZFA70 135611366 IC50 = 626 nM T85943 C0J3BN 135678111 IC50 > 50000 nM T85943 CPV59N 135685787 Ki > 4000 nM T85943 CDM07Y 135692621 IC50 = 9100 nM T85943 CU29YK 135750268 IC50 = 75 nM T85943 C1OE3C 135836172 IC50 = 64 nM T85943 CX4ZB3 135863110 IC50 > 30000 nM T85943 CYDM01 135891431 IC50 = 0.6 nM T85943 CJV08H 135897884 IC50 = 4.9 nM T85943 C4K3XL 135897887 IC50 < 0.5 nM T85943 C93QJC 135897888 IC50 = 0.83 nM T85943 CX6JV7 135897894 IC50 = 2.2 nM T85943 C5QUL0 135897897 IC50 < 0.5 nM T85943 CLV7Y8 135897900 IC50 = 0.61 nM T85943 CFJZ14 135897904 IC50 = 3.9 nM T85943 CT2UV5 135897905 IC50 = 1.7 nM T85943 CG3UZ1 135927974 Ki > 1000 nM T85943 CTJ7R1 135934758 IC50 = 32000 nM T85943 CF1PS8 135934877 Ki > 4000 nM T85943 CIPA79 135937899 IC50 > 10000 nM T85943 C12UDA 135947972 IC50 = 43 nM T85943 CN42ZS 135947973 IC50 = 15 nM T85943 CF8AO3 135947974 IC50 = 54 nM T85943 CW08GJ 135947976 IC50 = 131 nM T85943 CJN7E2 135947978 IC50 = 120 nM T85943 CFKH34 135947979 IC50 = 55 nM T85943 CTRL59 135976660 Ki > 4000 nM T85943 C0G1UL 135998453 Ki = 1240 nM T85943 C9W6BT 136002660 IC50 = 5400 nM T85943 CD9CT6 136002661 IC50 = 1840 nM T85943 C4T9KZ 136002662 IC50 = 930 nM T85943 CLY6I0 136023326 IC50 = 38000 nM T85943 CL2UH3 136023327 IC50 = 550000 nM T85943 C2R9NQ 136023328 IC50 = 1550000 nM T85943 CAWS49 136023329 IC50 = 500 nM T85943 C7WYX9 136023330 IC50 = 3700 nM T85943 C5XIE8 136026041 IC50 = 7700 nM T85943 C26ESH 136060555 IC50 > 50000 nM T85943 CVIC49 136069671 IC50 = 870 nM T85943 CIZ4K5 136088587 IC50 = 1500 nM T85943 CQ84IZ 136180335 Ki > 4000 nM T85943 CZ7EX0 136183413 IC50 = 1310 nM T85943 C2U0DL 136185991 IC50 = 2.1 ug.mL-1 T85943 CD48LY 136185992 IC50 = 1.25 ug.mL-1 T85943 CPE2B1 136185998 IC50 = 3 ug.mL-1 T85943 CR9XE0 136185999 IC50 = 0.9 ug.mL-1 T85943 C1I8LC 136186000 IC50 = 3.6 ug.mL-1 T85943 C40HWO 136186001 IC50 = 5 ug.mL-1 T85943 CK5VW8 136186003 IC50 = 1.2 ug.mL-1 T85943 C7V1YL 136186004 IC50 = 9 ug.mL-1 T85943 CJY3M8 136186005 IC50 = 0.6 ug.mL-1 T85943 CGP04W 136186009 IC50 = 12 ug.mL-1 T85943 CS5QE7 136186010 IC50 > 20 ug.mL-1 T85943 CDT7E4 136211077 IC50 > 100 nM T85943 CQM35B 136231164 IC50 > 10000 nM T85943 CX73ZW 136231169 Ki > 10000 nM T85943 CM63AX 136245248 Ki < 100 nM T85943 C5ZLF3 136254284 IC50 = 1200 nM T85943 CWT54E 136254285 IC50 > 10000 nM T85943 CXC69T 137321158 IC50 = 173 nM T85943 CE75QD 137321162 IC50 = 240 nM T85943 C3Z7BX 137355931 IC50 = 3 nM T85943 C25ERN 137631967 IC50 = 6.4 nM T85943 CZOD53 137633880 IC50 = 265 nM T85943 CI1E8V 137634241 IC50 = 156 nM T85943 C9S5ZG 137635614 Ki = 3000 nM T85943 C79XWZ 137636138 Ki > 100000 nM T85943 C7BJY5 137636807 IC50 = 112 nM T85943 C06JRX 137637094 IC50 = 5.7 nM T85943 C07CQL 137637848 Ki = 800 nM T85943 CQTF50 137641213 Ki = 2500 nM T85943 C36KUM 137642749 Ki = 2000 nM T85943 C7KQH8 137644946 Ki = 500 nM T85943 CO89DX 137649100 IC50 = 77 nM T85943 C1DK0P 137651391 IC50 = 6 nM T85943 CINE03 137652514 IC50 = 512 nM T85943 C28QUP 137652864 IC50 = 197 nM T85943 C71HKP 137655481 Ki = 6000 nM T85943 C0YP9H 137657483 Ki = 1500 nM T85943 CV5H3Z 137657932 IC50 = 3.9 nM T85943 C64GHK 137659108 Ki = 4700 nM T85943 C1XW3M 137659733 Ki = 5000 nM T85943 CSRI06 138547901 IC50 > 1000 nM T85943 CUXO19 138617501 IC50 > 1000 nM T85943 C63CUW 138857405 IC50 = 3 nM T85943 CRWA29 139030520 IC50 = 902.5 nM T85943 CO9P7G 145351804 IC50 > 1000 nM T85943 C6VB3O 145925651 IC50 >= 5000 nM T85943 C29XUO 145945978 IC50 > 1000 nM T85943 C4HB8M 145949394 IC50 = 61 nM T85943 C65YWX 145964882 IC50 = 3600 nM T85943 CHC3T0 145965031 IC50 > 10000 nM T85943 CP92ZF 145965329 IC50 = 1100 nM T85943 C9HXI4 145966620 IC50 = 1000 nM T85943 CQE9M5 145966810 IC50 = 800 nM T85943 C1EH6C 145967078 IC50 = 7200 nM T85943 CWJ12M 145969155 IC50 = 93 nM T85943 CGW5S1 145969844 IC50 = 8300 nM T85943 CB8R3A 145970271 IC50 > 10000 nM T85943 C40VIL 145972979 IC50 = 890 nM T85943 CQBY19 145974023 IC50 > 10000 nM T85943 C4X7CT 145977420 IC50 > 10000 nM T85943 CLA57T 145978300 IC50 > 10000 nM T85943 CXV58W 145980843 Ki = 120 nM T85943 C5EBY0 145980898 Ki = 190 nM T85943 C0WQO8 145981153 Ki = 50 nM T85943 C2ACE9 145982279 Ki = 3.5 nM T85943 C9YKF5 145986311 Ki = 840 nM T85943 CUO9P8 145989101 Ki = 300 nM T85943 C7Y3TI 145989362 Ki = 33 nM T85943 C6B7LV 145990977 Ki = 74 nM T85943 C5JY6O 145991326 Ki = 17 nM T85943 CQR73Y 145991889 Ki = 60 nM T85943 C5Q1NA 145992041 Ki = 3.5 nM T85943 CM3T6U 145993898 Ki = 23 nM T85943 CC2AQ0 154573782 IC50 = 3 nM T85943 COZA72 155415442 IC50 = 2 nM T85943 C82YKF 155415443 IC50 = 9 nM T85943 CQC20K 155415472 IC50 = 3 nM T85943 C3Y0WX 155415493 IC50 = 5 nM T85943 CL98BI 155415495 IC50 = 5 nM T85943 C4GZ7D 155415496 IC50 = 6 nM T85943 C8UOT3 155415499 IC50 = 3 nM T85943 CHKX30 155415500 IC50 > 3330 nM T85943 C94HAT 155415504 IC50 = 940 nM T85943 CYD73X 155415508 IC50 = 8 nM T85943 CMJZ23 155415509 IC50 = 6 nM T85943 C09YSN 155415512 IC50 = 5 nM T85943 CK2W1A 155415513 IC50 = 22 nM T85943 CNF0X5 155415516 IC50 = 79 nM T85943 CD2B5T 155415517 IC50 = 4 nM T85943 CJ0DO6 155415524 IC50 = 4010 nM T85943 CK8Y9I 155415561 IC50 = 14 nM T85943 C59VKN 155415568 IC50 = 6 nM T85943 CGM4U0 155415583 IC50 = 1010 nM T85943 C1XD0Z 155432267 IC50 = 8 nM T85943 C6P9DC 155432378 IC50 = 33 nM T85943 C9F2GQ 155432379 IC50 = 121 nM T85943 CK52YN 155432383 IC50 = 226 nM T85943 C1RWE8 155432590 IC50 = 7 nM T85943 CP9TU0 155432614 IC50 > 10000 nM T85943 CF27EG 155511610 IC50 = 897 nM T85943 C4PT8S 155511865 IC50 = 5.3 nM T85943 C0AN1O 155512752 IC50 = 804 nM T85943 C2MD1Q 155513187 IC50 > 10000 nM T85943 CM9V5R 155513533 Ki = 0.851 nM T85943 CA0TO6 155514385 IC50 = 97 nM T85943 C86HPW 155518524 IC50 = 8800 nM T85943 C3VTM7 155519139 IC50 = 383 nM T85943 C3NA2I 155519537 IC50 = 123 nM T85943 C2XY3V 155519623 IC50 = 1210 nM T85943 CHX98P 155522217 Ki = 0.925 nM T85943 C3E9NR 155527921 IC50 = 3580 nM T85943 C54ARD 155532371 IC50 = 15100 nM T85943 C16YZS 155534423 Ki = 0.785 nM T85943 C3LC9I 155536820 IC50 = 2511.89 nM T85943 C3V4LG 155538413 IC50 = 209 nM T85943 D00ERW 44444843 Ki > 1936 nM T85943 D00GVV 5329155 IC50 = 4920 nM T85943 D00HVA 11624601 Ki > 1900 nM T85943 D00TBD 10461815 IC50 = 6000 nM T85943 D00TVY 44300176 IC50 = 5500 nM T85943 D00YCU 667662 IC50 > 50000 nM T85943 D01FWD 606669 IC50 > 50000 nM T85943 D01GNF 10301426 Ki = 500 nM T85943 D01IDD 1036901 Ki = 1900 nM T85943 D01IZN 44312289 IC50 = 1600 nM T85943 D01JJR 447522 IC50 = 10 nM T85943 D01VFR 4708 IC50 = 73 nM T85943 D01YWE 25207521 IC50 > 50000 nM T85943 D02BXJ 46864270 IC50 = 4 nM T85943 D02HOG 5287488 IC50 = 900000 nM T85943 D02IYN 5287555 IC50 = 2200 nM T85943 D02RTS 311 IC50 > 40000000 nM T85943 D02SRA 44312288 IC50 = 2100 nM T85943 D02TIO 447524 IC50 = 450 nM T85943 D02XKJ 5328466 IC50 > 50000 nM T85943 D03EHM 24905142 IC50 = 14 nM T85943 D03GQI 1049055 Ki = 4300 nM T85943 D03MUZ 17759555 IC50 = 19900 nM T85943 D03NCK 5287443 IC50 = 120 nM T85943 D03NPX 447077 IC50 = 24.5 nM T85943 D03OKV 9844320 IC50 = 96 nM T85943 D04QUI 2250919 Ki = 500 nM T85943 D05FXD 44478401 IC50 = 1.14 nM T85943 D05GYO 5287515 IC50 = 437 nM T85943 D05NKG 16760286 IC50 = 316.23 nM T85943 D05PTT 5281792 IC50 = 26000 nM T85943 D05YQC 447534 IC50 = 4400000 nM T85943 D06CYG 44300143 IC50 = 800 nM T85943 D06EZQ 5324595 IC50 = 350 nM T85943 D06HVH 54613583 IC50 > 10000 nM T85943 D06KSF 9549300 IC50 > 400000 nM T85943 D06LJL 9916282 IC50 = 3000 nM T85943 D06QUQ 5311381 IC50 = 19.95 nM T85943 D06QWO 14824655 IC50 > 10 ug.mL-1 T85943 D06WGX 9549184 IC50 = 9050 nM T85943 D06ZCX 10455969 IC50 > 100000 nM T85943 D07ADX 54764565 IC50 = 4330 nM T85943 D07ERV 44312580 IC50 = 540 nM T85943 D07HBR 5287461 IC50 = 2300000 nM T85943 D07LYJ 1075248 Ki = 5400 nM T85943 D07OAT 456214 IC50 = 240 nM T85943 D07RQB 44419363 IC50 = 5200 nM T85943 D07SRX 9797919 IC50 = 7000 nM T85943 D08JNG 867 IC50 > 40000000 nM T85943 D08RZB 11153014 IC50 < 2 nM T85943 D08WEV 821478 Ki = 2900 nM T85943 D09DVB 44312287 IC50 = 1000 nM T85943 D09QKH 1097674 Ki = 2000 nM T85943 D09RYV 9911652 IC50 = 3210000 nM T85943 D09WNM 5289215 IC50 = 1200000 nM T85943 D0A1CM 5281855 IC50 = 300 nM T85943 D0A2LX 44312363 IC50 = 130 nM T85943 D0A4XJ 5289418 IC50 = 10600 nM T85943 D0A5MG 1094114 Ki = 4100 nM T85943 D0AJ4T 5287463 IC50 = 80000 nM T85943 D0AY0F 70698427 IC50 > 10000 nM T85943 D0B4PI 44312309 IC50 = 2900 nM T85943 D0BS6R 9549183 IC50 = 70 nM T85943 D0BU6T 354471 IC50 = 3500 nM T85943 D0BW4G 10907042 IC50 > 30000 nM T85943 D0C2GE 67161540 IC50 = 33 nM T85943 D0C9KC 10850934 IC50 > 100000 nM T85943 D0CE3R 5312137 IC50 = 73 nM T85943 D0CM6T 11314340 Ki = 13000 nM T85943 D0D1FK 5287465 IC50 = 500000 nM T85943 D0D3RL 44517649 IC50 = 7600 nM T85943 D0D5EW 5311104 IC50 = 16.8 nM T85943 D0D6DH 10125830 IC50 > 50000 nM T85943 D0D6MH 11617559 IC50 > 16000 nM T85943 D0D8OY 25210550 IC50 = 7000 nM T85943 D0D8ZN 1728080 Ki = 1000 nM T85943 D0D9PD 11656591 IC50 = 3.9 nM T85943 D0E7VO 59627005 IC50 = 18.2 nM T85943 D0EE6A 6398883 IC50 > 10000 nM T85943 D0EH6L 10360970 IC50 > 100000 nM T85943 D0EW3L 5281222 IC50 = 65000 nM T85943 D0G3SZ 6918469 IC50 = 8.3 ug.mL-1 T85943 D0GW4Q 5330524 IC50 = 66.3 nM T85943 D0H1OK 11562302 Ki = 11 nM T85943 D0H2CM 135565635 IC50 = 1400 nM T85943 D0H3XF 135463744 IC50 = 10000 nM T85943 D0IR6U 5494425 IC50 > 8000 nM T85943 D0J3LR 11634725 Ki > 4000 nM T85943 D0J4RY 1103113 Ki = 1300 nM T85943 D0K2YG 5328512 IC50 > 50000 nM T85943 D0KS2T 447518 IC50 = 9 nM T85943 D0L0HG 766949 IC50 > 10000 nM T85943 D0L3FK 5289419 IC50 = 11000 nM T85943 D0L4HJ 5330462 IC50 = 280 nM T85943 D0L4NP 5287544 IC50 = 0.25 nM T85943 D0LP2M 1021453 Ki = 900 nM T85943 D0M5RA 447537 IC50 = 3900000 nM T85943 D0M9QM 5327820 IC50 = 501.19 nM T85943 D0MI2W 11643573 IC50 = 6400 nM T85943 D0N8TQ 10401956 IC50 = 126 nM T85943 D0OG1Q 2049536 IC50 = 7943.28 nM T85943 D0OH3J 5330526 IC50 = 9.03 nM T85943 D0OZ2S 11785878 IC50 = 120 nM T85943 D0P2QG 1113004 Ki = 1000 nM T85943 D0P3JW 447700 IC50 = 43 nM T85943 D0P5ST 18455703 IC50 = 12000 nM T85943 D0Q2UZ 44312307 IC50 = 1800 nM T85943 D0Q3NG 11715520 Ki > 1900 nM T85943 D0Q7TO 6419766 Ki = 81 nM T85943 D0R1PD 447527 IC50 = 2000 nM T85943 D0R2WK 16038120 EC50 > 1000 nM T85943 D0R7BX 75791 IC50 = 200000 nM T85943 D0S1KJ 5328733 IC50 = 8 nM T85943 D0S3FW 44422490 IC50 = 5500 nM T85943 D0S7IE 11658882 Ki > 1900 nM T85943 D0S9LT 12793 IC50 = 3500000 nM T85943 D0T0YI 378 IC50 = 1000000 nM T85943 D0TC1E 447523 IC50 = 4 nM T85943 D0U5KF 5287550 IC50 = 300000 nM T85943 D0U7BY 971 IC50 > 40000000 nM T85943 D0U8UH 447532 IC50 = 3600000 nM T85943 D0UN9O 3385203 IC50 >= 10000 nM T85943 D0W7LW 44312308 IC50 = 1500 nM T85943 D0XS9E 5330535 IC50 > 30000 nM T85943 D0Y0BK 11524144 IC50 = 2 nM T85943 D0Y1SR 11844351 IC50 = 6 nM T85943 D0YE1X 9927943 IC50 > 10000 nM T85943 D0YZ7H 9797370 IC50 = 185 nM T85943 D0Z7GH 5330525 IC50 = 16.3 nM T85943 D0ZH1U 2051 IC50 = 2700 nM T68230 C5TR0L 132213490 IC50 = 3400 nM T68230 CZF35N 132213510 IC50 = 11000 nM T68230 CL4O7S 132213544 IC50 = 3200 nM T68230 C2EKZ5 132213594 IC50 = 760 nM T68230 C4X6JM 132213664 IC50 = 480 nM T68230 C3GFA9 132213677 IC50 = 1500 nM T68230 CRC3H4 132213711 IC50 = 1100 nM T68230 C9O7GU 132213775 IC50 = 1800 nM T68230 CM67WC 132213878 IC50 = 37000 nM T68230 C3R4HZ 132213912 IC50 = 920 nM T68230 CU94VK 132213922 IC50 = 690 nM T68230 C39LDP 132213961 IC50 = 17000 nM T68230 C5FG3K 132214001 IC50 = 860 nM T68230 CT25BP 132214054 IC50 > 100000 nM T68230 C1ROB2 132214070 IC50 = 23000 nM T68230 C2UR9C 132214083 IC50 = 2600 nM T68230 CT03JX 132214086 IC50 = 5300 nM T68230 C1R7CV 132214131 IC50 = 580 nM T68230 CIR6A9 132214222 IC50 = 6300 nM T68230 C4JRU5 132214241 IC50 = 3000 nM T68230 C6UAG3 132214357 IC50 = 31000 nM T68230 C5U0ME 132214417 IC50 > 100000 nM T68230 CJ7O6E 132214420 IC50 = 2400 nM T68230 CK5V8M 132214443 IC50 = 1100 nM T68230 C8MYQ9 132214492 IC50 = 8100 nM T68230 CT40BX 132214508 IC50 = 2100 nM T68230 CLN9T7 132214550 IC50 = 860 nM T68230 CV32LW 132218314 IC50 = 18000 nM T37539 C89WEN 25138688 IC50 = 24760 nM T37539 C58KRC 25138689 IC50 = 37700 nM T37539 C1DR0M 25138690 IC50 = 470 nM T37539 CO7KP8 25138849 IC50 = 5480 nM T37539 C0HX5I 25138850 IC50 = 6220 nM T37539 CSLT92 25138851 IC50 = 530 nM T37539 CW19FC 25139009 IC50 = 43000 nM T37539 C3ZO7Q 25139010 IC50 = 7480 nM T37539 C47XHY 25139011 IC50 = 1730 nM T37539 CZ91HW 25139165 IC50 = 230 nM T37539 CR59FL 25139166 IC50 = 1760 nM T37539 C5Z6HB 25139167 IC50 = 9830 nM T37539 CPLV74 25139317 IC50 = 45000 nM T37539 CE89CW 25140005 IC50 = 148330 nM T37539 CCW7I6 25140006 IC50 = 85000 nM T37539 CJ6D5N 25140159 IC50 = 125160 nM T37539 C27JVH 25140160 IC50 = 192670 nM T37539 CT3WD8 25140161 IC50 = 115850 nM T37539 CN6FT9 25140162 IC50 = 132320 nM T37539 CM09ZX 25140311 IC50 = 16000 nM T37539 CXRZ31 25140312 IC50 = 40850 nM T37539 C0NHT2 25140313 IC50 = 10400 nM T37539 C1KW2X 25140314 IC50 = 7650 nM T37539 CKG81Y 25140456 IC50 = 21060 nM T37539 CG5I3E 25140457 IC50 = 2600 nM T37539 C7K4UY 25140458 IC50 = 8850 nM T37539 CA7T8N 25140598 IC50 = 1100 nM T37539 C0M4QL 25140599 IC50 = 3700 nM T37539 C78QKJ 25140600 IC50 = 1000 nM T37539 C3H5PZ 25140735 IC50 = 400 nM T37539 C4P2XC 25140736 IC50 = 900 nM T37539 CYE47Q 25140737 IC50 = 4300 nM T37539 C90XJG 25140892 IC50 = 7130 nM T37539 C9KM2N 25140893 IC50 = 73250 nM T37539 CE0R7Z 25140894 IC50 = 122570 nM T37539 C9FJ6P 44588730 IC50 = 683330 nM T37539 CG04MH 44588731 IC50 = 550000 nM T37539 C7CXU9 53317637 IC50 = 130 nM T37539 CKE7U4 53318681 IC50 = 820 nM T37539 CFUB60 53322630 IC50 = 70 nM T37539 CMYR56 53323963 IC50 = 1120 nM T95302 D0X9PF 9941379 Ki = 17 nM T95302 CL04VQ 910537 Ki = 141000 nM T95302 C0DA9X 2163781 Ki = 18000 nM T95302 CK4YT2 2817655 Ki = 100000 nM T95302 CB9A2M 2852098 Ki = 14000 nM T95302 CWZ1O2 6918780 EC50 = 210 nM T95302 CY60AZ 6918813 EC50 = 1900 nM T95302 C2BQE1 6918814 Ki = 280 nM T95302 CK83QR 6918844 Ki = 560 nM T95302 CLV3C7 6918849 IC50 = 24 nM T95302 C5U7CS 6918850 Ki = 540 nM T95302 C0Q5JL 6918851 EC50 = 850 nM T95302 CRG04O 6918857 Ki = 950 nM T95302 COS6C1 9808720 EC50 = 230 nM T95302 CM02VS 9808801 IC50 = 430 nM T95302 CM3Y5H 9893728 IC50 > 10000 nM T95302 CZ5E2C 9915636 Ki = 1000 nM T95302 CCL2T8 9915813 EC50 = 4400 nM T95302 C15DES 9924916 Ki = 18000 nM T95302 C7V8AE 9946241 Ki = 29000 nM T95302 C6L4VG 9946358 Ki = 20000 nM T95302 CX5CU3 9958649 Ki = 11 nM T95302 C97MRJ 9960253 Ki = 1200 nM T95302 CMU31X 9968756 Ki = 25000 nM T95302 C5F3QU 9969456 Ki = 18000 nM T95302 CLXA58 10025669 Ki = 36000 nM T95302 C8KI2R 10033237 Ki = 27 nM T95302 CZ78WX 10077258 IC50 = 250 nM T95302 C8MCA1 10077773 Ki = 2200 nM T95302 CSQ60B 10108894 Ki = 35000 nM T95302 C6LVA2 10109225 Ki = 4900 nM T95302 CG1K8Y 10122170 EC50 = 79 nM T95302 CF81WV 10132207 Ki = 27000 nM T95302 C0PVS9 10134057 Ki = 58000 nM T95302 CC0ZT7 10137615 Ki = 11000 nM T95302 CO69QN 10146211 EC50 = 170 nM T95302 C03AKT 10155513 Ki = 89000 nM T95302 CPRS08 10157774 Ki = 5200 nM T95302 CXF16O 10158674 Ki = 7300 nM T95302 C97IHD 10159196 Ki = 23000 nM T95302 CAB06U 10177247 Ki = 12000 nM T95302 COJ1M5 10178845 Ki = 4300 nM T95302 CV2QX0 10180932 Ki = 34000 nM T95302 C78FGS 10188529 EC50 = 850 nM T95302 C1HMR6 10200110 Ki = 16000 nM T95302 CFZ5I6 10210964 IC50 = 34 nM T95302 C8PA3J 10211466 Ki = 1400 nM T95302 CWJ5I0 10225762 Ki = 34000 nM T95302 CTO7I8 10232787 Ki = 1200 nM T95302 CSNY06 10257242 IC50 = 660 nM T95302 C6Y1ER 10257541 Ki = 9800 nM T95302 C2AL7S 10260053 Ki = 880 nM T95302 CEC2M0 10269187 Ki = 23000 nM T95302 C6T2MU 10270570 Ki = 19000 nM T95302 CX29KB 10282847 IC50 = 31 nM T95302 C4SCW2 10283036 Ki = 420 nM T95302 CSDX25 10291370 Ki = 930 nM T95302 CX97KY 10292084 Ki = 25000 nM T95302 CU17RB 10293285 Ki = 267000 nM T95302 CV3ZJ5 10304463 Ki = 920 nM T95302 CU13DH 10304547 IC50 = 64 nM T95302 C1E3PC 10304776 IC50 = 54 nM T95302 CT9AR6 10325955 Ki = 700 nM T95302 CPL02I 10463896 IC50 > 1000 nM T95302 CTEB92 10483153 EC50 = 1000 nM T95302 CBPX36 10864861 EC50 = 271 nM T95302 CGIC31 10918643 IC50 > 10000 nM T95302 CAL9N7 11017471 EC50 = 1004 nM T95302 C7IJV5 11038873 EC50 = 10000 nM T95302 CHOS10 11061068 EC50 = 127 nM T95302 CO2U6S 11156852 Ki = 2300 nM T95302 CYLZ82 11179871 Ki = 560 nM T95302 C3V7DK 11180881 Ki = 720 nM T95302 CHC51K 11181804 Ki = 240 nM T95302 CTO68V 11191792 Ki = 1050 nM T95302 CJO5T1 11192466 Ki = 290 nM T95302 CD5SG6 11215758 Ki = 600 nM T95302 CF7VQ4 11226756 Ki = 1400 nM T95302 CWLJ34 11237444 Ki = 5.3 nM T95302 C1T3VM 11249545 Ki = 5.9 nM T95302 C7AD6W 11272524 Ki = 144 nM T95302 CP9S6F 11273288 EC50 = 450 nM T95302 C4JA5I 11284919 Ki = 1760 nM T95302 CLS9A8 11295934 Ki = 70 nM T95302 CJ7OT2 11296600 Ki = 270 nM T95302 C2PU1F 11296732 Ki = 990 nM T95302 C8PKU9 11318528 Ki = 91 nM T95302 CS7K4R 11341045 Ki = 18 nM T95302 CU6Y1Z 11341046 Ki = 26 nM T95302 CAL3F9 11364326 Ki = 21 nM T95302 CLHF89 11365127 Ki = 77 nM T95302 C5D1TY 11375764 Ki = 2.1 nM T95302 CX8EJ9 11410616 Ki = 305 nM T95302 CMR57W 11433304 Ki = 44 nM T95302 CHD05I 11443753 Ki = 360 nM T95302 C8LN5W 11477853 Ki = 36 nM T95302 C3J4CM 11752660 Ki = 50 nM T95302 CH7TQ6 11753695 IC50 = 83.9 nM T95302 CXBR04 11785639 Ki = 230 nM T95302 C2UO9X 11785893 Ki = 350 nM T95302 C2SHV7 11786860 Ki = 590 nM T95302 C0OIV9 11813437 EC50 = 9400 nM T95302 CT4EC3 11966875 IC50 > 10000 nM T95302 CI9W3G 15953833 EC50 = 2400 nM T95302 CAT74W 15953838 IC50 = 1410 nM T95302 C54MIL 16007264 Ki = 500 nM T95302 C6XS3N 16007285 Ki = 170 nM T95302 CYW0B8 16038315 Ki = 2100 nM T95302 C4N0VF 16046215 Ki = 1000 nM T95302 CX68DN 16049796 IC50 = 0.1 nM T95302 CPTO16 16132144 EC50 = 8.1 nM T95302 C4NZ3C 16725559 EC50 = 1600 nM T95302 C25XZF 17880880 Ki = 256000 nM T95302 CFNQ06 23635107 Ki = 180 nM T95302 CHU29W 23635235 Ki = 340 nM T95302 CWL5K4 23635236 Ki = 340 nM T95302 CVFQ41 23635237 Ki = 320 nM T95302 CBW09O 23653113 Ki = 13000 nM T95302 C8KO9M 23661656 Ki = 990 nM T95302 CK2Q5J 24180592 Ki = 600 nM T95302 C7SMW5 24180646 Ki = 850 nM T95302 CU19BT 24740419 Ki = 1200 nM T95302 CTC05L 24740653 Ki = 710 nM T95302 CD90WZ 24740655 Ki = 520 nM T95302 CUPD43 24741624 Ki = 86 nM T95302 C5TA3W 24774358 IC50 = 790 nM T95302 CO4JK2 24774437 IC50 > 10000 nM T95302 CMB27G 24774521 IC50 = 120 nM T95302 C2TAK6 24774601 IC50 > 10000 nM T95302 C2A1SX 24848995 Ki = 1200 nM T95302 C1EN7W 24857886 IC50 = 450 nM T95302 CB9M3F 24873537 Ki = 240 nM T95302 CG9AV5 25058412 Ki = 970 nM T95302 C4SH1P 25211670 Ki = 540 nM T95302 C4HK6C 42630327 IC50 = 1905.46 nM T95302 CU4S6X 44157099 EC50 = 85 nM T95302 CBG73U 44158097 EC50 = 2500 nM T95302 CIOF26 44158168 EC50 = 1.6 nM T95302 C53LJK 44158169 IC50 = 1.1 nM T95302 C9UD8I 44158336 IC50 = 22 nM T95302 CF6PT4 44158337 EC50 = 0.3 nM T95302 CHKI60 44265225 Ki > 1000000 nM T95302 CXN2R4 44265309 Ki = 43000 nM T95302 C3EJ1R 44265312 Ki = 38000 nM T95302 CWPT03 44265315 Ki = 173000 nM T95302 CJ1M6N 44265347 Ki = 28000 nM T95302 CEQ6K7 44265351 Ki = 45000 nM T95302 CSL48C 44265374 Ki = 4100 nM T95302 C97AIK 44265472 Ki = 47000 nM T95302 C6DZ4W 44265473 Ki = 83000 nM T95302 CLE96R 44265479 Ki = 74000 nM T95302 CV8GX6 44265487 Ki = 36000 nM T95302 C2CPG9 44265489 Ki = 150000 nM T95302 CLP5G3 44265496 Ki = 2500 nM T95302 C51TPY 44265586 Ki > 1000 nM T95302 CH5WM7 44265588 Ki > 1000 nM T95302 CT89LY 44265589 Ki = 74000 nM T95302 CZS3C7 44265590 Ki = 130000 nM T95302 C3YKG9 44265591 Ki = 56000 nM T95302 C74SBD 44265625 Ki > 1000 nM T95302 CRQ92O 44265626 Ki > 1000 nM T95302 CT2S8I 44265639 Ki = 8700 nM T95302 C18JZD 44265656 Ki = 184000 nM T95302 CD8UC0 44265662 Ki > 1000 nM T95302 C6OU7D 44265665 Ki > 1000 nM T95302 CC28FH 44265672 Ki = 15000 nM T95302 CSK9V6 44265674 Ki > 1000 nM T95302 CS46LN 44265675 Ki = 125000 nM T95302 C9E0TB 44265681 Ki = 221000 nM T95302 CCGI15 44265707 Ki = 15000 nM T95302 CION54 44265708 Ki = 60000 nM T95302 C9CM8W 44265711 Ki = 37000 nM T95302 CPUO61 44265713 Ki = 50000 nM T95302 CP1E6X 44265715 Ki = 6600 nM T95302 CRFQ64 44265719 Ki = 95000 nM T95302 CXUI50 44265722 Ki = 200000 nM T95302 CVEG42 44265727 Ki > 1000 nM T95302 CC4S8V 44265739 Ki > 1000 nM T95302 CG1CH0 44265748 Ki > 1000 nM T95302 C82FPN 44265749 Ki = 42000 nM T95302 C05MIH 44265751 Ki = 1000000 nM T95302 CP82FI 44265757 Ki > 1000 nM T95302 CE6A0Z 44265759 Ki > 1000 nM T95302 CPE83Q 44269189 EC50 = 3900 nM T95302 CCP5L2 44269214 EC50 = 2700 nM T95302 CN5TI2 44269217 EC50 = 2100 nM T95302 CBW0I1 44275650 EC50 = 33 nM T95302 C5OHC4 44277696 IC50 = 13300 nM T95302 CU8PH5 44293516 IC50 > 1000 nM T95302 C7DZ1Q 44293599 IC50 > 1000 nM T95302 C57HNX 44307979 IC50 > 10000 nM T95302 C8LZV7 44308004 IC50 > 10000 nM T95302 CFP7W8 44308044 IC50 > 10000 nM T95302 C79WRA 44308214 IC50 > 10000 nM T95302 CT76SR 44308215 IC50 > 10000 nM T95302 CQ59BO 44320339 Ki = 3981.07 nM T95302 C27QTD 44322795 EC50 = 560 nM T95302 C3XED9 44322868 EC50 = 1.01 nM T95302 C8P1HE 44322869 Ki = 3100 nM T95302 CEDS20 44323020 EC50 = 640 nM T95302 CW49BO 44323234 Ki = 140 nM T95302 C8BID0 44325926 IC50 = 557 nM T95302 CD9ER8 44343341 Ki = 26 nM T95302 CCLF38 44347081 Ki = 4900 nM T95302 CT5V4X 44347082 Ki = 4900 nM T95302 C0QW9K 44347105 Ki = 4800 nM T95302 CWK01G 44347106 Ki = 2700 nM T95302 C4Y2SW 44347107 Ki = 20 nM T95302 C60PGA 44347110 Ki = 5000 nM T95302 CUEZ31 44347119 Ki = 130 nM T95302 CT03JB 44347219 EC50 = 530 nM T95302 COD7W0 44347220 Ki = 65 nM T95302 CNP94O 44347221 Ki = 150 nM T95302 CBE37A 44347277 Ki = 24 nM T95302 CIZ30K 44347294 Ki = 720 nM T95302 C2YQM4 44347330 Ki = 7000 nM T95302 CX0Z1Y 44347331 Ki = 140 nM T95302 CAKI17 44347344 Ki = 0.09 nM T95302 CEIM86 44347370 EC50 = 0.22 nM T95302 CS5ID0 44347378 Ki = 2400 nM T95302 CDN35X 44347379 Ki = 2500 nM T95302 CENG52 44347433 Ki = 18 nM T95302 CW1JY7 44347434 EC50 = 4.2 nM T95302 C24GLU 44347435 EC50 = 19 nM T95302 C7U2KM 44347838 IC50 = 94 nM T95302 CK6FH3 44347927 IC50 = 200 nM T95302 C58SIF 44348144 EC50 > 10000 nM T95302 C0F1EA 44348183 IC50 = 97000 nM T95302 CC41MG 44348199 EC50 > 10000 nM T95302 CRSW34 44348200 EC50 > 10000 nM T95302 C6E7SA 44349019 EC50 > 3000 nM T95302 C2QW1I 44364160 EC50 = 390 nM T95302 CLMA12 44366081 IC50 = 0.027 nM T95302 C2DHN5 44366155 EC50 = 45 nM T95302 CYD6R3 44366171 EC50 = 530 nM T95302 CO7U1L 44366182 IC50 = 4.6 nM T95302 CL4CY1 44366187 EC50 = 390 nM T95302 C9JN3L 44366213 EC50 = 17 nM T95302 C36FMV 44366215 IC50 = 0.031 nM T95302 CS27ZR 44366381 EC50 = 0.2 nM T95302 CQCP89 44387680 EC50 = 82 nM T95302 CD8HL0 44392514 Ki = 17000 nM T95302 CE21OM 44392535 Ki = 18000 nM T95302 C3IHV4 44393417 Ki = 16000 nM T95302 C2J1ML 44393418 Ki = 14000 nM T95302 CQ3L0D 44393421 Ki = 8200 nM T95302 C9C7SD 44393430 Ki = 102000 nM T95302 C47HVD 44393441 Ki = 17000 nM T95302 C1OG5U 44393450 Ki = 94000 nM T95302 CK5D8I 44394079 Ki = 260 nM T95302 CVUQ61 44395681 Ki = 1000 nM T95302 CLT7X4 44396002 Ki = 730 nM T95302 C8D2RU 44396986 EC50 = 1980 nM T95302 C6Z9BD 44396987 IC50 = 1020 nM T95302 CZ2C9L 44397028 Ki = 470 nM T95302 CDZ3O4 44397030 Ki = 480 nM T95302 C9V2RU 44397198 Ki = 920 nM T95302 C9CF7N 44397220 IC50 = 1080 nM T95302 CXQ0M6 44397281 Ki = 1200 nM T95302 CPM68W 44397283 Ki = 1400 nM T95302 CX07ID 44397304 Ki = 1900 nM T95302 C7TNB6 44397410 IC50 = 840 nM T95302 C6F0QR 44397455 IC50 = 40 nM T95302 C49FRZ 44397461 IC50 = 1400 nM T95302 CL6KA2 44397652 IC50 = 1200 nM T95302 CJ36UT 44400660 Ki = 730 nM T95302 C5NJQ2 44400812 Ki = 2300 nM T95302 CC8SI2 44400813 Ki = 350 nM T95302 CAR95M 44400863 Ki = 680 nM T95302 C2VI7C 44400864 Ki = 300 nM T95302 C61RQJ 44400934 Ki = 350 nM T95302 C2IJZ5 44400935 Ki = 160 nM T95302 C1QM4Y 44401310 EC50 = 880 nM T95302 CM9W3D 44401520 EC50 = 710 nM T95302 CIQH79 44401522 EC50 = 340 nM T95302 CDSM37 44401524 EC50 = 760 nM T95302 CVN78D 44401528 EC50 = 360 nM T95302 C4R9XD 44401530 EC50 = 300 nM T95302 C5AQD6 44401585 EC50 = 2400 nM T95302 CRMV98 44408154 IC50 = 190 nM T95302 CIWX60 44408155 IC50 = 200 nM T95302 COG72Y 44408173 IC50 = 170 nM T95302 C3CQ4J 44408189 EC50 = 460 nM T95302 CW08ZJ 44408190 EC50 = 280 nM T95302 CNWJ27 44408252 IC50 = 150 nM T95302 CH68SP 44408253 EC50 = 3600 nM T95302 CCFV91 44408275 EC50 = 400 nM T95302 CZ3YG9 44408276 EC50 = 620 nM T95302 CAFP51 44408286 EC50 = 340 nM T95302 CR8HZ7 44408287 EC50 = 400 nM T95302 COC7D2 44408388 EC50 = 1200 nM T95302 C48WZD 44410802 Ki = 2000 nM T95302 C43IKV 44410803 Ki = 910 nM T95302 C7IYH9 44415417 Ki = 1200 nM T95302 C4G2BZ 44417555 IC50 = 209 nM T95302 C32QEO 44418413 IC50 = 0.4 nM T95302 C7FEU6 44418420 IC50 = 0.8 nM T95302 CZW07E 44418421 EC50 > 10000 nM T95302 CLQG83 44418430 EC50 > 10000 nM T95302 C8VG1S 44418431 EC50 > 10000 nM T95302 C3HPI5 44418437 IC50 = 0.5 nM T95302 CMD5N2 44418438 IC50 = 0.1 nM T95302 CQE30X 44422937 IC50 = 390 nM T95302 C14FZP 44422938 IC50 > 2000 nM T95302 CE0H3Y 44422957 IC50 > 10000 nM T95302 C6H0NU 44422958 IC50 > 10000 nM T95302 C7I0KW 44422959 IC50 > 10000 nM T95302 C46XOB 44422960 IC50 > 10000 nM T95302 CNM90E 44422961 IC50 > 10000 nM T95302 C2K3BL 44422962 IC50 > 10000 nM T95302 C3E6VO 44422994 EC50 = 770 nM T95302 CHU7G0 44422996 EC50 > 1500 nM T95302 C2LQW9 44422997 EC50 = 82 nM T95302 CJM09S 44422998 EC50 = 670 nM T95302 CI9HF1 44422999 EC50 = 2.5 nM T95302 CXH5F8 44423009 IC50 = 250 nM T95302 C3VOD0 44423010 EC50 = 50 nM T95302 C7UI3W 44423011 IC50 = 2700 nM T95302 CI05BD 44423012 IC50 > 10000 nM T95302 C5EJ3P 44423013 IC50 > 10000 nM T95302 C2NR7G 44423014 EC50 = 1500 nM T95302 CV3TL5 44423015 EC50 = 270 nM T95302 CN5RD6 44431510 EC50 > 10000 nM T95302 CF3H8A 44431511 IC50 = 2900 nM T95302 CVB07O 44431512 IC50 = 123 nM T95302 CY80GN 44431513 IC50 = 87 nM T95302 COCE51 44431515 EC50 = 3.3 nM T95302 CV62SP 44432932 Ki = 880 nM T95302 CL3ZR1 44432964 Ki = 5900 nM T95302 C0L4NV 44432966 Ki = 1600 nM T95302 CKX7P2 44433264 Ki = 250 nM T95302 CZU4D1 44433294 Ki = 1300 nM T95302 CW8B6E 44433439 Ki = 380 nM T95302 C8Z1IM 44434561 Ki = 408000 nM T95302 C5C6IA 44434562 Ki = 240 nM T95302 C6KPV5 44434568 Ki = 360 nM T95302 C2K9TI 44434570 Ki = 13000 nM T95302 CBC27H 44434581 Ki = 12000 nM T95302 C51NSB 44434584 Ki = 3400 nM T95302 CF2S6P 44434587 Ki = 3200 nM T95302 CQ81UI 44434592 Ki = 23000 nM T95302 CP2A4G 44434595 Ki = 55000 nM T95302 CT20IC 44434597 Ki = 33000 nM T95302 CC1H3U 44434598 Ki = 13000 nM T95302 CH17AO 44434599 Ki = 12000 nM T95302 CAID38 44434600 Ki = 11000 nM T95302 CGN1P8 44434601 Ki = 10000 nM T95302 CDV61Y 44434603 Ki = 31000 nM T95302 CZPC57 44434605 Ki = 91000 nM T95302 C5DT7Q 44434611 Ki = 12000 nM T95302 C3MS2D 44434613 Ki = 681000 nM T95302 C5A1GF 44434614 Ki = 25000 nM T95302 CN4D2E 44434616 Ki = 13000 nM T95302 C1B5RV 44434621 Ki = 35000 nM T95302 C5TMA6 44434625 Ki = 279000 nM T95302 C9XG2K 44434631 Ki = 353000 nM T95302 CY2C7G 44434632 Ki = 10000 nM T95302 CQ94YK 44434633 Ki = 85000 nM T95302 CM1NA8 44434634 Ki = 56000 nM T95302 C93NCL 44434635 Ki = 20000 nM T95302 CZ8TO1 44434636 Ki = 4600 nM T95302 CQ06DV 44434637 Ki = 7900 nM T95302 C3T4JG 44434639 Ki = 19000 nM T95302 C0SM2J 44434647 Ki = 46000 nM T95302 C9GIF5 44434648 Ki = 8000 nM T95302 C15MAF 44434650 Ki = 8000 nM T95302 CWD27I 44434651 Ki = 6700 nM T95302 C6X8WB 44434652 Ki = 2200 nM T95302 CWU74N 44434653 Ki = 28000 nM T95302 CXN0M3 44434654 Ki = 5400 nM T95302 CM0VZ8 44434655 Ki = 8700 nM T95302 CP0V1N 44434656 Ki = 17000 nM T95302 CV5Y3N 44434657 Ki = 24000 nM T95302 CVC93Q 44434658 Ki = 34000 nM T95302 CWE1V4 44434659 Ki = 102000 nM T95302 C5WR3A 44434661 Ki = 20000 nM T95302 CJ27QL 44434662 Ki = 4600 nM T95302 C6US7A 44434663 Ki = 5100 nM T95302 C4ZD1B 44434664 Ki = 159000 nM T95302 C03NKU 44434665 Ki = 54000 nM T95302 CJ2AT0 44434666 Ki = 8000 nM T95302 CF41SX 44434682 Ki = 21000 nM T95302 C9IWD4 44434683 Ki = 20000 nM T95302 CJ03PB 44434684 Ki = 3800 nM T95302 CIH0Z6 44434685 Ki = 2100 nM T95302 C4POB8 44434686 Ki = 31000 nM T95302 C1GFE6 44434687 Ki = 29000 nM T95302 C3J7WI 44434688 Ki = 3200 nM T95302 C9Y0BM 44434689 Ki = 40000 nM T95302 CH6LA5 44434690 Ki = 3200 nM T95302 CPRE40 44434691 Ki = 8300 nM T95302 C9O8LX 44434692 Ki = 11000 nM T95302 CE2Z3V 44434693 Ki = 9500 nM T95302 C31LUY 44434694 Ki = 12000 nM T95302 C9C4BN 44434695 Ki = 7200 nM T95302 CF3JX5 44434696 Ki = 36000 nM T95302 CM51SC 44434697 Ki = 9600 nM T95302 CA2FQ4 44434698 Ki = 6700 nM T95302 CTC18P 44434699 Ki = 85000 nM T95302 CQT85W 44434700 Ki = 8900 nM T95302 C8BQ7C 44434701 Ki = 12000 nM T95302 CV2QW3 44434702 Ki = 16000 nM T95302 C9IY3A 44434703 Ki = 15000 nM T95302 CF8J2P 44434704 Ki = 4400 nM T95302 CH7QD5 44434706 Ki = 10000 nM T95302 CT4FO2 44434707 Ki = 2200 nM T95302 C9E4PO 44434709 Ki = 9100 nM T95302 C7LUV2 44434713 Ki = 5000 nM T95302 CR70OD 44434714 Ki = 49000 nM T95302 CA1BF3 44434715 Ki = 278000 nM T95302 C0N4CY 44434753 Ki = 23000 nM T95302 CS1KG4 44434754 Ki = 7600 nM T95302 C2JHP0 44434757 Ki = 266000 nM T95302 CZ43DV 44434758 Ki = 18000 nM T95302 C50PIJ 44434759 Ki = 96000 nM T95302 CKAQ59 44434760 Ki = 5200 nM T95302 CALF38 44434761 Ki = 97000 nM T95302 C17HCY 44434762 Ki = 4300 nM T95302 CX75CS 44434763 Ki = 11000 nM T95302 CNB68V 44434764 Ki = 5200 nM T95302 CZ0R9M 44434765 Ki = 15000 nM T95302 CU9C0K 44434766 Ki = 3900 nM T95302 C8IHB1 44434767 Ki = 21000 nM T95302 C27KYV 44434768 Ki = 7200 nM T95302 CEM27N 44434769 Ki = 22000 nM T95302 CB7A2G 44434770 Ki = 83000 nM T95302 C0Y3IG 44434771 Ki = 21000 nM T95302 CNL2T3 44434772 Ki = 4900 nM T95302 CUW4Y6 44434778 Ki = 5500 nM T95302 CH8WT0 44434780 Ki = 44000 nM T95302 CL9K2D 44434781 Ki = 18000 nM T95302 CJ12GC 44434782 Ki = 7700 nM T95302 CFBX46 44434785 Ki = 6900 nM T95302 C0KB8P 44434787 Ki = 9100 nM T95302 C0M2VI 44434790 Ki = 15000 nM T95302 CH3UV8 44434794 Ki = 17000 nM T95302 C10VDG 44434797 Ki = 8300 nM T95302 CWN02S 44434799 Ki = 28000 nM T95302 C0X1MK 44434821 Ki = 6100 nM T95302 CU1ON8 44434828 Ki = 16000 nM T95302 CBHU73 44434839 Ki = 21000 nM T95302 C20UIF 44434841 Ki = 11000 nM T95302 CA7P5L 44434843 Ki = 24000 nM T95302 CBL2D7 44434845 Ki = 2600 nM T95302 CYE25C 44434847 Ki = 37000 nM T95302 CWE0J6 44434848 Ki = 6400 nM T95302 CB39YP 44434849 Ki = 32000 nM T95302 C0ZV6S 44434850 Ki = 17000 nM T95302 C4U6LJ 44434851 Ki = 9700 nM T95302 CA4M3C 44434853 Ki = 555000 nM T95302 CVGW87 44434854 Ki = 4800 nM T95302 C3G5QO 44434855 Ki = 1700 nM T95302 C2JET5 44434856 Ki = 6600 nM T95302 C2M5VB 44434857 Ki = 22000 nM T95302 CS30KD 44434858 Ki = 176000 nM T95302 C7S1OK 44434859 Ki = 52000 nM T95302 C3AVB5 44434860 Ki = 10000 nM T95302 CZQI93 44434861 Ki = 40000 nM T95302 CC0U5Y 44434862 Ki = 11000 nM T95302 CWTI58 44434863 Ki = 18000 nM T95302 CFOM13 44434864 Ki = 37000 nM T95302 CL97ID 44434865 Ki = 16000 nM T95302 CW93VX 44434867 Ki = 49000 nM T95302 CN36OD 44434868 Ki = 23000 nM T95302 CI09FJ 44434870 Ki = 10000 nM T95302 CZE48F 44434872 Ki = 18000 nM T95302 CXTV37 44434880 Ki = 9100 nM T95302 CQ45JU 44434884 Ki = 8700 nM T95302 CZ8H3M 44435220 Ki = 12000 nM T95302 CPM80E 44441633 EC50 = 640 nM T95302 CD25AP 44441636 EC50 = 480 nM T95302 CQL07M 44441637 EC50 = 1100 nM T95302 CEHV41 44441639 EC50 = 630 nM T95302 C5D6YN 44441641 EC50 = 222 nM T95302 CP4TW0 44441642 EC50 = 662 nM T95302 CDC3R8 44441643 EC50 = 380 nM T95302 CU6ZN4 44441644 EC50 = 250 nM T95302 CNS4O1 44441645 EC50 = 684 nM T95302 CRL83D 44441646 EC50 = 1760 nM T95302 C7EQ6Z 44441647 EC50 = 527 nM T95302 CHSV38 44441648 EC50 = 2950 nM T95302 C3MIO4 44441681 EC50 = 977 nM T95302 CT3J4B 44441684 EC50 = 888 nM T95302 C3YRT9 44441685 EC50 = 1117 nM T95302 CCS5T3 44441687 EC50 = 1980 nM T95302 C08BMY 44448479 EC50 = 1233 nM T95302 C0C7KI 44448590 EC50 = 166.7 nM T95302 CQHR95 44448629 EC50 = 101.6 nM T95302 C78XDT 44448631 EC50 = 455 nM T95302 C8H1UT 44448660 IC50 = 129.4 nM T95302 C63APB 44456219 Ki = 530 nM T95302 CE0P7K 44456222 Ki = 800 nM T95302 C5CIX6 44562287 Ki = 950 nM T95302 CU92FG 44562414 Ki = 330 nM T95302 CPSC21 44562440 Ki = 1800 nM T95302 CQ0I1K 44562460 Ki = 540 nM T95302 CD3T1I 44577060 Ki = 1100 nM T95302 C6FI8E 44577062 Ki = 110 nM T95302 CJ6GZ3 44577063 Ki = 400 nM T95302 CWOK70 44577090 Ki = 1100 nM T95302 C4FSH3 44577091 Ki = 67 nM T95302 CF8PL1 44577092 Ki = 13 nM T95302 CM6X5S 44577093 Ki = 34 nM T95302 CGTV08 44577094 Ki = 390 nM T95302 CEJ96P 44577510 EC50 = 44 nM T95302 CRSQ61 44577514 IC50 = 760 nM T95302 C6Y1BS 44577515 IC50 = 130 nM T95302 C8B1WR 44577520 IC50 = 340 nM T95302 C3NSW7 44577523 IC50 > 2000 nM T95302 CWFB17 44583567 EC50 = 1.9 nM T95302 CJB6H0 46203215 EC50 = 20000 nM T95302 CD3E4C 46885323 EC50 > 20000 nM T95302 CE4SF8 46885368 EC50 = 1430 nM T95302 CHPS01 46885417 EC50 > 20000 nM T95302 C4SVE1 46885480 EC50 = 960 nM T95302 COU5X2 46885482 EC50 > 20000 nM T95302 C90ABZ 46885558 EC50 > 14000 nM T95302 C0MI3C 46885560 EC50 > 11100 nM T95302 C0Y9NF 46885711 EC50 = 5190 nM T95302 C3O5BR 46885712 EC50 = 3600 nM T95302 CG6XN0 46885759 EC50 = 1800 nM T95302 CK8D6G 46885760 EC50 > 5810 nM T95302 C0C8GN 46885761 EC50 = 3500 nM T95302 CY30PG 46885815 EC50 = 17800 nM T95302 CWN89S 46885863 EC50 = 15000 nM T95302 C8UTI7 46885907 EC50 = 6410 nM T95302 CFC5L1 46885972 EC50 = 3640 nM T95302 C29LQB 46919520 IC50 = 122.7 nM T95302 C1EMQ2 49861348 EC50 = 1980 nM T95302 C9QU3G 49862375 EC50 = 490 nM T95302 CPZI97 49862377 EC50 = 1000 nM T95302 CY7R2T 49862378 IC50 = 1100 nM T95302 C7GA4I 49862425 IC50 = 2800 nM T95302 C0QD9I 51346770 Ki = 388 nM T95302 C30PGL 51346771 Ki = 1532 nM T95302 CBQN64 52918026 IC50 = 850 nM T95302 CG5TJ0 53240339 IC50 = 300 nM T95302 C6GET3 54582029 IC50 = 1000 nM T95302 CQ7O3U 54584301 IC50 = 1400 nM T95302 C8PIL3 54584302 EC50 = 1400 nM T95302 CN6F2C 54586246 IC50 = 1300 nM T95302 CEU0M6 54587278 EC50 = 210 nM T95302 CTSB57 56850936 Ki = 58 nM T95302 C1U2DB 56851057 Ki = 46 nM T95302 C2WAO4 57634921 Ki = 5.1 nM T95302 C4VT5C 57634925 Ki = 4.3 nM T95302 CKW2T0 57646411 Ki = 0.47 nM T95302 C8F5XG 57646441 Ki = 1.6 nM T95302 CH1LU3 58777892 Ki = 280 nM T95302 C73SKU 70682946 EC50 = 410 nM T95302 CBY2K9 70683600 EC50 = 1000 nM T95302 C0O6QG 70685712 EC50 = 1400 nM T95302 CPJ08L 70688853 Ki = 3 nM T95302 CU86WQ 70689887 EC50 = 920 nM T95302 CB2X0A 70689888 EC50 = 1900 nM T95302 CE28CX 70691332 IC50 = 0.09 nM T95302 C81JGS 70692049 EC50 = 45 nM T95302 C97FOR 70696210 EC50 = 1400 nM T95302 C2O7TA 71449047 EC50 = 190 nM T95302 CH0F4A 71449048 IC50 = 10 nM T95302 C1JN2M 71449119 EC50 = 1800 nM T95302 CJPX32 71449204 EC50 = 510 nM T95302 CKCN10 71452720 IC50 = 940 nM T95302 CEB0P9 71452732 Ki = 700 nM T95302 CV0J8X 71452824 EC50 = 840 nM T95302 CN4EJ2 71452825 EC50 = 340 nM T95302 CW8OE1 71452826 EC50 = 2000 nM T95302 CY16AM 71454518 Ki = 10000 nM T95302 CPX03G 71456219 EC50 = 880 nM T95302 C07WXP 71456220 IC50 = 73 nM T95302 CNRV69 71456245 IC50 = 690 nM T95302 CU17GR 71458055 Ki = 4000 nM T95302 C6YR0U 71458117 IC50 > 10000 nM T95302 CJ52CU 71459938 IC50 = 3100 nM T95302 CU2A1J 71461601 EC50 = 5000 nM T95302 CECQ16 71461657 Ki = 260 nM T95302 C24GWM 71461662 Ki = 12000 nM T95302 CZ94CM 71461730 EC50 = 6.01 nM T95302 CYA8G1 71717886 EC50 = 250 nM T95302 CV8K5U 73345513 EC50 = 1.8 nM T95302 C4IAM6 73345514 Ki > 4800 nM T95302 C1A5SK 73345616 IC50 = 1500 nM T95302 CI0DV9 73345617 EC50 = 0.99 nM T95302 CD1NE3 73345618 EC50 > 500 nM T95302 CYMH60 73347015 Ki = 16 nM T95302 CZ91TE 73347138 EC50 = 0.37 nM T95302 CK46SP 73347139 IC50 = 10 nM T95302 CX9LF8 73347140 EC50 = 0.29 nM T95302 C4SR8Z 73348617 IC50 = 2 nM T95302 CS4I5R 73350057 EC50 = 3.3 nM T95302 CMLR03 73350220 EC50 = 0.031 nM T95302 C3EF0P 73351617 Ki = 14 nM T95302 CKWH98 73351727 EC50 = 0.45 nM T95302 C1L7HK 73353100 Ki = 1 nM T95302 CJL0D3 73353101 EC50 = 210 nM T95302 C8C0LW 73353205 EC50 = 0.23 nM T95302 CGVC68 73353206 IC50 = 24 nM T95302 CK2X0G 73353271 IC50 = 21 nM T95302 CK23FW 73354573 Ki = 22 nM T95302 CIEJ89 73354618 Ki = 17 nM T95302 C0ISQ4 73354708 EC50 = 1.6 nM T95302 CJS25D 73354709 EC50 = 1 nM T95302 C7OT4D 73354780 EC50 = 69 nM T95302 C17PEL 73356313 IC50 = 1.24 nM T95302 CP1S3T 90664642 EC50 = 2700 nM T95302 CR7OX0 90664763 EC50 = 3300 nM T95302 C1KS2F 101043843 EC50 = 10.1 nM T95302 CI8PR4 118718122 EC50 = 49 nM T95302 CCL46X 118718855 IC50 > 10000 nM T95302 CK6FL5 118718881 IC50 = 141 nM T95302 C8ME0B 118735099 IC50 = 636 nM T95302 CK17XF 118735100 IC50 = 167 nM T95302 C1O7GU 118735101 IC50 = 70.3 nM T95302 CBTC79 118735102 IC50 = 37.3 nM T95302 C1O3GL 118735103 IC50 = 137 nM T95302 C65WMB 122184498 EC50 = 7 nM T95302 CH9L8O 122184499 EC50 = 60 nM T95302 CAQ17N 122184571 IC50 = 16.8 nM T95302 CK48WX 122184572 EC50 = 1060 nM T95302 CF9PO7 122184573 IC50 = 27.7 nM T95302 C3FBZ9 122184574 IC50 = 5 nM T95302 CCP0X7 122184575 EC50 = 1560 nM T95302 C7OBX1 122184576 EC50 = 446 nM T95302 CU73AF 122184577 IC50 = 95 nM T95302 CGB7F4 122184578 IC50 = 13 nM T95302 CB7HZ8 122184579 EC50 = 460 nM T95302 C9HE4L 122184580 EC50 > 2000 nM T95302 C9MJT7 122184581 IC50 = 91 nM T95302 C20NAY 122184582 IC50 = 35.2 nM T95302 CH1B8W 122184631 IC50 = 6.33 nM T95302 CLXB63 122184632 IC50 = 1670 nM T95302 CIJ14O 122184633 IC50 = 6.66 nM T95302 CDSR31 122184634 IC50 = 592 nM T95302 CL28BX 122184635 EC50 = 1.1 nM T95302 CYOR02 122184636 IC50 = 39.7 nM T95302 C09LFS 122184637 EC50 = 239 nM T95302 C5CDX9 122184638 IC50 = 388 nM T95302 C64BPZ 122184639 IC50 = 159 nM T95302 CEDT39 122184640 EC50 = 838 nM T95302 CLB43S 122184641 EC50 = 62.52 nM T95302 CN4L5U 122184908 EC50 = 1680 nM T95302 CG0U7B 122184909 IC50 = 1510 nM T95302 CZ4HW7 122184910 EC50 = 0.8 nM T95302 C6KW7J 122184911 EC50 = 1450 nM T95302 CK3VM5 122184912 EC50 = 818 nM T95302 C0AFH9 122184913 EC50 = 1520 nM T95302 CNBA05 122184914 IC50 = 257 nM T95302 CJNF06 137631599 IC50 = 281.84 nM T95302 CW9P1D 137633115 IC50 = 36 nM T95302 CF2NA9 137633806 EC50 = 109.7 nM T95302 CTD90C 137634090 EC50 > 100000 nM T95302 CPL59T 137635422 EC50 = 298.7 nM T95302 CM1H6A 137636428 EC50 > 3000 nM T95302 CU4KL7 137636677 IC50 = 6606.93 nM T95302 CVC3Q2 137636965 IC50 = 16218.1 nM T95302 CK2CZ3 137637026 EC50 = 916 nM T95302 CME01A 137637283 EC50 = 0.93 nM T95302 C6TKX9 137637656 EC50 = 375.2 nM T95302 CMJ4I7 137637705 IC50 = 0.42 nM T95302 C2FEA6 137638725 IC50 > 1000 nM T95302 CH17TL 137638778 EC50 = 137 nM T95302 CZ74WU 137639140 EC50 > 100000 nM T95302 CKR14I 137639770 EC50 = 8.1 nM T95302 CHB9X0 137640703 IC50 = 4168.69 nM T95302 CBL5Z9 137641157 IC50 = 707.95 nM T95302 CCPD94 137641398 IC50 = 812.83 nM T95302 CGP0V3 137643023 EC50 > 3000 nM T95302 CAT50J 137643076 IC50 > 1000 nM T95302 C5R2TI 137643266 IC50 = 254 nM T95302 CE0YF4 137643385 EC50 > 3000 nM T95302 C68AYB 137644225 EC50 > 3000 nM T95302 CJ1I7B 137645567 IC50 > 1000 nM T95302 CKES17 137646333 IC50 > 100000 nM T95302 CT18GM 137646617 IC50 = 11220.18 nM T95302 CV5RX4 137647009 EC50 > 3000 nM T95302 CY7K4J 137647538 IC50 = 1122.02 nM T95302 C10VFY 137648144 EC50 > 3000 nM T95302 CSF97J 137649543 EC50 > 3000 nM T95302 CIV6Z7 137649910 EC50 > 3000 nM T95302 C7I9CK 137651025 EC50 > 100000 nM T95302 CF3VP0 137651074 EC50 = 16 nM T95302 CH62TM 137653176 EC50 > 3000 nM T95302 CF5Z2W 137653739 EC50 = 1 nM T95302 CKX3Q9 137653925 IC50 = 7079.46 nM T95302 CMO01K 137655905 IC50 = 4073.8 nM T95302 CKL0Y8 137656033 EC50 > 3000 nM T95302 C5WHL4 137656521 EC50 = 752.3 nM T95302 C5FI6X 137657633 IC50 = 330 nM T95302 COS0A1 137658158 IC50 = 8511.38 nM T95302 CS1PR7 137659394 IC50 > 1000 nM T95302 CHB32J 137659790 IC50 = 25118.86 nM T95302 CQ7S0L 137659949 EC50 > 100000 nM T95302 C2XLI7 137660671 IC50 = 758.58 nM T95302 C98FVD 137660993 IC50 = 58.88 nM T95302 C4CFP9 137661893 EC50 >= 809 nM T95302 CCZ72V 137662147 EC50 = 635 nM T95302 C2WC5J 145948876 EC50 = 20 nM T95302 CUC3S2 145948912 EC50 = 73 nM T95302 C8D7OM 145964017 EC50 = 170 nM T95302 CCK75J 145964837 EC50 = 18 nM T95302 CHU51B 145966490 EC50 = 14 nM T95302 CJO1Y6 145966716 EC50 = 560 nM T95302 C9RA7Q 145967155 IC50 = 21 nM T95302 CICD84 145971389 EC50 = 2 nM T95302 C97DEG 145971673 IC50 > 1000 nM T95302 CEV4F6 145972289 IC50 > 1000 nM T95302 C9NRU8 145973779 IC50 = 20 nM T95302 CYD0J5 145973975 EC50 = 96 nM T95302 CR2NQ5 145975465 EC50 = 140 nM T95302 CKP26E 145976444 IC50 = 12 nM T95302 C7UJ8Q 145976863 EC50 = 1.9 nM T95302 CMS17N 145977650 IC50 > 1000 nM T95302 C0S1IN 145980719 EC50 = 37 nM T95302 CF34MX 145988152 EC50 > 1000 nM T95302 C7WF3R 145989222 EC50 = 433 nM T95302 C50ZLS 145990599 IC50 = 37 nM T95302 C10FUX 145994325 IC50 > 5000 nM T95302 C5S4PT 24858479 IC50 = 560 nM T95302 CA83CB 24858481 IC50 = 38 nM T95302 CR08PO 24858629 IC50 = 58 nM T95302 D00TSX 11672424 IC50 = 2.3 nM T95302 D00VYC 44400370 Ki > 500 nM T95302 D01HTX 11707715 IC50 = 70 nM T95302 D01VMU 44445082 EC50 = 570 nM T95302 D02JVA 44408515 IC50 = 2.3 nM T95302 D02MPZ 11535237 IC50 = 100 nM T95302 D03AZC 25078192 Ki = 0.84 nM T95302 D04BOG 11629290 EC50 > 10000 nM T95302 D04YZZ 44445083 EC50 = 23 nM T95302 D05LLI 11498895 IC50 = 1.4 nM T95302 D05WNC 11520823 IC50 = 44 nM T95302 D05XRI 44400401 Ki > 500 nM T95302 D06RTP 11700730 IC50 = 2.2 nM T95302 D07DWH 44400402 Ki > 500 nM T95302 D07IBF 44400322 Ki > 500 nM T95302 D07SFD 44408443 IC50 = 68 nM T95302 D07UXW 44408400 IC50 = 220 nM T95302 D08DND 44445084 IC50 = 520 nM T95302 D09OMI 44400400 Ki > 500 nM T95302 D09PDT 24774519 IC50 = 210 nM T95302 D09UUC 46877881 Ki = 990 nM T95302 D09XCH 44400371 Ki > 500 nM T95302 D0A8ME 44400398 Ki > 500 nM T95302 D0B9NH 44408399 IC50 = 3060 nM T95302 D0C7VI 44400369 Ki > 500 nM T95302 D0GN9K 24774602 IC50 > 10000 nM T95302 D0L1MJ 11700739 EC50 = 200 nM T95302 D0M4EF 11593084 IC50 = 110 nM T95302 D0N6KO 9938402 IC50 = 326 nM T95302 D0P4GI 11629326 IC50 = 10 nM T95302 D0QW4A 24774356 IC50 > 1000 nM T95302 D0R0BY 44400320 Ki = 42.19 nM T95302 D0U5KM 11093672 EC50 = 3.9 nM T95302 D0VD7R 44408408 EC50 = 850 nM T95302 D0W1SM 44408413 EC50 = 300 nM T95302 D0WG8P 44400321 Ki = 239.3 nM T95302 D0WI8M 44445085 IC50 = 17 nM T95302 D0X1YL 25078242 Ki = 62.11 nM T95302 D0XQ5U 24774438 IC50 = 230 nM T95302 D0YB7F 92432 EC50 = 1.48 nM T95302 D0ZD3M 44400399 Ki > 500 nM T58992 D00KHM 16362 IC50 = 3760 nM T58992 D00UYE 4058 IC50 > 10000 nM T58992 D01KQA 5311304 Ki = 240 nM T58992 D02NSF 5284604 IC50 = 45 nM T58992 D02RXG 6918287 Ki = 693 nM T58992 D03DIG 5284371 IC50 > 9300 nM T58992 D03SKD 5284603 EC50 = 4000 nM T58992 D03YVO 5361917 Ki = 501.19 nM T58992 D04JEE 4946 EC50 > 5011.87 nM T58992 D04JHN 5284570 Ki = 38 nM T58992 D05GKD 33741 Ki > 10000 nM T58992 D05VIL 5284594 Ki = 9.3 nM T58992 D09OJQ 4095 IC50 = 1090 nM T58992 D09ZXR 11250029 EC50 > 10000 nM T58992 D0CQ0Z 33630 Ki = 1714 nM T58992 D0CS2F 3955 EC50 = 156 nM T58992 D0D7KC 5488548 Ki = 5.012 nM T58992 D0E1WI 3345 IC50 = 187 nM T58992 D0G8NN 119570 Ki > 10000 nM T58992 D0PG8O 5360515 EC50 = 4.4 nM T58992 D0T3HY 5359272 IC50 = 2.9 nM T58992 D0WE3O 5288826 EC50 = 15.6 nM T58992 D0X3FX 5284596 Ki = 19 nM T58992 D0X9RG 5361092 Ki = 12 nM T58992 D00HBR 5486554 IC50 = 23 nM T58992 D03PJU 62156 Ki = 3.28 nM T58992 D06ENM 66553195 EC50 = 2800 nM T58992 D06EXA 128563 Ki = 3990 nM T58992 D07TQN 179340 EC50 = 8000 nM T58992 D07YHM 44129648 Ki = 122 nM T58992 D09ALE 60768 Ki > 1000 nM T58992 D0LI1C 44469321 IC50 > 10000 nM T58992 D0N1HW 5311200 Ki > 10000 nM T58992 D0Q3PD 54732242 Ki = 0.91 nM T58992 D0R0EF 24772484 IC50 = 0.28 nM T58992 D0RN6V 9865223 Ki = 1000 nM T58992 D0T0ZW 11667832 EC50 = 1.8 nM T58992 D0V5WL 443363 EC50 = 1.03 nM T58992 D0W4YO 16131448 Ki > 1000 nM T58992 D0C2QF 9906198 Ki = 0.312 nM T58992 D0M1YN 5311194 Ki > 400 nM T58992 D0N1RG 9805452 Ki = 0.18 nM T58992 D00ACC 9844019 Ki > 400 nM T58992 D06DZI 107780 Ki > 10000 nM T58992 D08YUP 9950038 EC50 = 0.7 nM T58992 D0G1YN 9826770 IC50 = 3.4 nM T58992 D0K5KL 119029 EC50 = 0.12 nM T58992 D0LX5D 5487663 EC50 = 1 nM T58992 D0M7BW 3505 IC50 > 10000 nM T58992 D0W8TS 9898185 IC50 = 29 nM T58992 C21VAX 1223 IC50 = 1.5 nM T58992 CAG0J1 5523 Ki = 9.4 nM T58992 C5H9CN 9287 Ki > 10000 nM T58992 CZC17M 9669 Ki = 49 nM T58992 C6E8DS 62513 Ki > 10000 nM T58992 CBGO28 70419 Ki = 2946 nM T58992 CX5R6B 71420 IC50 = 123 nM T58992 CYKE31 104920 IC50 > 10000 nM T58992 C3CU5L 107772 EC50 = 371.54 nM T58992 C9NJK8 114876 Ki = 3713 nM T58992 CQYC47 121999 Ki = 9.1 nM T58992 CDM08R 124716 Ki = 23 nM T58992 CFZ4W6 127914 IC50 > 1000 nM T58992 CB8Y9H 134131 Ki = 33 nM T58992 CO26HG 134377 Ki = 5.2 nM T58992 CM2H7V 152430 Ki = 3100 nM T58992 C0UZ5G 159564 Ki = 0.3 nM T58992 C9B1MS 159966 IC50 = 46000 nM T58992 CM5I3Z 161271 Ki > 26000 nM T58992 CVL3Z7 190901 IC50 > 1000 nM T58992 C4LEU1 191408 Ki > 10000 nM T58992 C3HB4V 416359 IC50 > 10000 nM T58992 CR45EB 644177 Ki = 6690 nM T58992 C3VFW0 715222 IC50 = 10000 nM T58992 C6BDH3 780684 EC50 = 7800 nM T58992 C8H0KW 1009511 EC50 = 100 nM T58992 C4U2MZ 1044308 EC50 = 100 nM T58992 C6B0TP 1121183 EC50 = 2000 nM T58992 CX8KH4 2297178 EC50 = 200 nM T58992 CAO06Q 2796048 IC50 > 10000 nM T58992 CLXC53 3000341 Ki = 2884.03 nM T58992 CAQ2J0 3034396 Ki = 60.26 nM T58992 C2TAD3 3036289 Ki = 2500 nM T58992 CLB7W5 3037886 Ki = 140 nM T58992 CH0Z2R 3037926 Ki = 0.58 nM T58992 C5HDK8 3041260 Ki = 77.3 nM T58992 C8OHF0 3081578 Ki = 9.8 nM T58992 CMKU43 3086068 Ki = 9.7 nM T58992 C19ESC 3086114 IC50 = 6.99 nM T58992 CJ6D8N 3342390 Ki = 1088 nM T58992 CC3DM1 3955796 EC50 = 300 nM T58992 CXO48E 4353400 EC50 = 300 nM T58992 C0LRX8 4491165 Ki = 0.3 nM T58992 CY7LK9 4491166 Ki = 3.4 nM T58992 CANE93 4545429 Ki = 24 nM T58992 C14LHW 5172692 EC50 = 200 nM T58992 CKLG29 5244802 Ki > 10000 nM T58992 C2O3TW 5282407 IC50 = 3630 nM T58992 CJX28Y 5311003 Ki = 1.7 nM T58992 CLW4B1 5311340 Ki = 8647 nM T58992 CN4V2F 5320438 Ki = 8400 nM T58992 C6HY1P 5361918 Ki = 501.19 nM T58992 C9XZY4 5362396 Ki = 0.02 nM T58992 C2HPQ4 5462505 Ki = 65.8 nM T58992 CV3K5Y 5484197 Ki = 58 nM T58992 C17RBP 5486940 Ki = 13.3 nM T58992 CH7EM4 5487533 IC50 = 818 nM T58992 CJ7IE6 5487695 Ki = 272 nM T58992 C2OU8T 5489400 IC50 = 37000 nM T58992 C41JIC 5490373 EC50 = 190 nM T58992 CCMZ86 5491688 Ki = 0.25 nM T58992 CZ4TM3 5492619 Ki = 4410 nM T58992 CI7L4R 5492830 Ki = 4520 nM T58992 C9LJ2K 5493351 Ki = 2.62 nM T58992 CJQN51 6438353 Ki = 1.8 nM T58992 C5AL8S 6445230 EC50 = 74.1 nM T58992 C5S8PV 6603740 Ki = 1000 nM T58992 CQML02 6603856 Ki = 422 nM T58992 CM6VF8 6734379 IC50 > 10000 nM T58992 C7A4HN 6916035 IC50 = 1.1 nM T58992 CFTO93 6918704 Ki = 166 nM T58992 CD49UV 9797246 Ki = 3791 nM T58992 C8ANR0 9801260 EC50 = 3.6 nM T58992 C5RNW7 9801830 IC50 > 10000 nM T58992 C3V7JB 9802297 Ki = 2.3 nM T58992 CPG57N 9803475 Ki > 400 nM T58992 C5GH0P 9804952 Ki = 450 nM T58992 CX7DO4 9806799 Ki = 578 nM T58992 C1TQM8 9809562 Ki = 2100 nM T58992 CVL4W8 9820950 Ki = 0.023 nM T58992 CJ72XV 9822639 Ki = 0.8 nM T58992 CXV1R9 9822756 IC50 = 4170 nM T58992 CG8XE0 9822764 Ki = 362 nM T58992 CE6NF9 9823363 IC50 > 10000 nM T58992 C9H5BP 9824054 Ki = 1010 nM T58992 C70KEP 9824565 Ki = 2998 nM T58992 CR54GJ 9824976 Ki = 3.5 nM T58992 CBXY90 9828569 Ki = 7.09 nM T58992 CW1T4D 9839245 Ki = 0.53 nM T58992 CX40CL 9840199 Ki = 1.259 nM T58992 C4QFZ6 9841259 EC50 = 7.2 nM T58992 CKVQ31 9843334 Ki = 3.7 nM T58992 C8JR0N 9843770 Ki = 184 nM T58992 C6Y7NA 9844540 Ki = 1665 nM T58992 CH06GL 9848989 IC50 = 0.9 nM T58992 CKD2H4 9848990 Ki = 1.15 nM T58992 CME87B 9849361 Ki = 0.1514 nM T58992 CBMN05 9865332 Ki = 2.2 nM T58992 CLQ6Z8 9866158 Ki = 3702 nM T58992 CL26PE 9866175 Ki = 6.2 nM T58992 C9BR6L 9871102 IC50 = 0.54 nM T58992 C51YLK 9871376 Ki = 1072 nM T58992 CPYK08 9887195 IC50 > 10000 nM T58992 C67GMC 9888235 Ki = 0.5 nM T58992 CB8G9J 9889993 Ki = 4.69 nM T58992 CJF8C2 9890982 EC50 = 0.75 nM T58992 C5BC4P 9902874 Ki > 10000 nM T58992 CUN81Q 9905249 Ki > 10000 nM T58992 C4X6PY 9909946 EC50 = 37 nM T58992 CB6C8L 9911987 Ki = 0.42 nM T58992 C26DMO 9928857 Ki = 33 nM T58992 CM3B5E 9932532 Ki = 1.2 nM T58992 C2U8XH 9932834 Ki = 3143 nM T58992 CYZW21 9932852 EC50 = 19 nM T58992 C9MK3B 9934232 Ki = 150385 nM T58992 CUBQ95 9937777 Ki = 906 nM T58992 CO7BI9 9940052 Ki = 70 nM T58992 C4FD7V 9947044 Ki = 480 nM T58992 CG9ER5 9947155 Ki > 2000 nM T58992 CF8UG9 9948520 Ki = 222 nM T58992 C5S3RH 9949205 Ki = 12.23 nM T58992 CUE9Z8 9951118 Ki = 15.85 nM T58992 CKNZ54 9951665 Ki = 0.3 nM T58992 COFT18 9951673 Ki = 1674 nM T58992 C3GXH0 9954388 Ki = 680 nM T58992 CT8C2X 9958643 Ki = 3204 nM T58992 CW02IS 9959144 Ki = 54 nM T58992 CI7GW2 9963195 Ki = 6.4 nM T58992 CE3CJ4 9969865 Ki > 2000 nM T58992 CC9ZU1 9973387 Ki = 1.48 nM T58992 C1B2JR 9976188 Ki > 1500 nM T58992 C2GI1Q 9984781 Ki = 38.22 nM T58992 CZA85S 9989078 IC50 = 1000 nM T58992 C2WJL0 9990996 Ki = 4507 nM T58992 CAGL19 9997843 Ki = 540 nM T58992 CN2F1U 10001960 IC50 = 0.63 nM T58992 CL9QS0 10004950 IC50 = 11.4 nM T58992 C9CP0Q 10005080 Ki = 110 nM T58992 C4Y8TH 10006938 IC50 = 0.35 nM T58992 CQ43EZ 10016044 Ki = 1.1 nM T58992 CV7R9F 10020040 Ki > 10000 nM T58992 C4N8YE 10020165 Ki > 10000 nM T58992 CL38DM 10021831 Ki = 103.4 nM T58992 C3J1VF 10022299 Ki = 5500 nM T58992 CHU1P6 10022640 IC50 = 144 nM T58992 C25DYT 10022859 Ki = 250 nM T58992 C0O9EM 10024658 IC50 > 10000 nM T58992 C85DQW 10026312 IC50 = 1.4 nM T58992 C96AWZ 10026663 IC50 > 1000 nM T58992 C60BIG 10028324 Ki = 13.9 nM T58992 C1PGE2 10031234 Ki = 0.79 nM T58992 C61SQU 10033525 IC50 = 11.9 nM T58992 C5KGS0 10041278 Ki = 134 nM T58992 C46PBM 10046193 Ki = 15 nM T58992 C5EGW6 10046467 IC50 = 21 nM T58992 CYI16O 10050608 IC50 = 55 nM T58992 CR16GC 10052760 IC50 = 312 nM T58992 C4CXP1 10053267 Ki = 3.4 nM T58992 C8WE1N 10055958 EC50 < 0.01 nM T58992 C8FLO9 10065022 Ki = 1760 nM T58992 CV37ET 10068300 IC50 = 1060 nM T58992 C8O4KB 10069687 Ki = 149 nM T58992 CS82YP 10071523 Ki = 6.5 nM T58992 CS3UK5 10074239 Ki = 12.5 nM T58992 CO8P3K 10076169 Ki = 1.8 nM T58992 CM34WV 10077545 Ki = 5 nM T58992 C3EBC8 10077792 Ki = 519 nM T58992 CKEW36 10078008 Ki = 137 nM T58992 CQVA98 10078468 Ki = 9.4 nM T58992 CPS53G 10080153 IC50 = 18.6 nM T58992 CL6N5H 10090388 Ki = 1.2 nM T58992 CZ5H9X 10093250 Ki = 0.025 nM T58992 C6UKP0 10094954 IC50 = 70 nM T58992 COU4D5 10099473 Ki = 109 nM T58992 C81PUC 10102939 IC50 = 1.63 nM T58992 C7YCF1 10109899 Ki = 975 nM T58992 CJNE19 10110916 Ki > 2000 nM T58992 C76MVA 10111186 Ki > 2000 nM T58992 C0PC9A 10113006 Ki = 35.9 nM T58992 CWEC34 10114637 Ki > 2000 nM T58992 CL5MY1 10116470 Ki = 24.1 nM T58992 CB4P7L 10116719 Ki = 103 nM T58992 C40BMF 10133108 Ki > 10000 nM T58992 CP1SO7 10134077 Ki > 10000 nM T58992 CEG0M4 10134217 Ki > 2000 nM T58992 C3ZTU0 10137134 Ki = 9784 nM T58992 C83KDV 10137876 Ki > 2000 nM T58992 C8E9KP 10139672 Ki > 2000 nM T58992 CVRZ09 10141332 Ki = 35.2 nM T58992 CT1B5J 10142188 Ki = 0.01 nM T58992 CKCW48 10143870 Ki = 17 nM T58992 CI3PJ6 10149623 Ki > 10000 nM T58992 CQGE97 10150001 Ki = 1856 nM T58992 CF85VW 10150089 Ki > 10000 nM T58992 C76SOW 10150260 Ki = 8344 nM T58992 CTO0N5 10158555 Ki = 33095 nM T58992 CWM2X6 10160920 Ki > 2000 nM T58992 C8ZA6U 10164835 Ki = 3.48 nM T58992 C67SZC 10171702 Ki = 10000 nM T58992 CDV15J 10172398 Ki = 634 nM T58992 CK5HG3 10179322 Ki = 2.9 nM T58992 CHC6K9 10179323 Ki = 1.8 nM T58992 C5RO6K 10182346 Ki > 2000 nM T58992 C2SP7U 10183838 Ki = 3.2 nM T58992 CUE8P2 10184592 Ki = 1.36 nM T58992 C2PTU7 10185016 Ki = 6.31 nM T58992 C2QF7B 10185709 Ki = 7.39 nM T58992 CNZL85 10193971 Ki = 9372 nM T58992 CN79QX 10194236 Ki = 6088 nM T58992 C12NGT 10199984 Ki > 2000 nM T58992 C85DFV 10201299 Ki = 4.6 nM T58992 CV1T7R 10202241 Ki > 2000 nM T58992 CZ4N2S 10205966 Ki = 352 nM T58992 C9ZCT0 10206319 Ki = 0.29 nM T58992 C1HP9A 10206324 Ki = 13.12 nM T58992 C31PWM 10206991 Ki = 2.62 nM T58992 C1J2WS 10207509 Ki = 49.53 nM T58992 C02IUS 10214859 Ki = 230 nM T58992 CYB0H9 10221539 IC50 > 1000 nM T58992 CRGJ86 10224456 IC50 > 10000 nM T58992 CM27FK 10225083 Ki = 368 nM T58992 C0I9TS 10226635 Ki = 20 nM T58992 C2XQR3 10227005 Ki = 32 nM T58992 C2MQS5 10227615 Ki = 0.93 nM T58992 CJW0B6 10228465 Ki = 0.38 nM T58992 CTF5Z8 10229655 Ki = 56 nM T58992 C6LQH4 10245350 Ki = 881 nM T58992 CKLA98 10246015 Ki = 150 nM T58992 CZ0C5T 10252647 Ki = 9111 nM T58992 CR4C1F 10253032 Ki = 2090 nM T58992 CLKQ39 10255149 EC50 = 22 nM T58992 C75HYP 10256020 Ki = 5.1 nM T58992 C4RX1A 10256503 Ki = 9.4 nM T58992 CH31DX 10267394 Ki > 10000 nM T58992 CWF4D9 10267592 Ki = 2.15 nM T58992 C58WLB 10273422 Ki = 0.39 nM T58992 C6YKB9 10273543 Ki = 500 nM T58992 C8PL7B 10274330 Ki > 2000 nM T58992 CO2M7L 10278214 Ki = 0.56 nM T58992 CUF17K 10279008 Ki = 49.01 nM T58992 C89KBW 10286378 Ki > 10000 nM T58992 CDP01X 10286440 Ki = 22410 nM T58992 C1FE9H 10286996 Ki = 9533 nM T58992 CJ14VU 10291377 Ki = 6532 nM T58992 CKO2I1 10297473 Ki = 0.74 nM T58992 CTG5B1 10300866 Ki = 924 nM T58992 CV0T3H 10301207 Ki = 1631 nM T58992 CF4VO2 10308746 Ki = 50 nM T58992 CU89JD 10314060 Ki > 10000 nM T58992 CFHC64 10315026 Ki = 22.4 nM T58992 CQD21X 10315939 Ki = 24.04 nM T58992 C7OXY2 10320559 IC50 = 3 nM T58992 CXN89V 10321082 IC50 = 34 nM T58992 C1ENR2 10323169 Ki = 538 nM T58992 CA4KJ5 10323346 EC50 = 1.2 nM T58992 C86PZN 10327545 Ki > 1000 nM T58992 CUJ0N2 10331735 Ki = 349 nM T58992 CH14KO 10334091 Ki = 29 nM T58992 C54WJL 10337395 Ki = 93 nM T58992 C91CEI 10339691 IC50 = 150 nM T58992 C63GNX 10342726 Ki = 177 nM T58992 CL38IN 10343372 Ki = 0.88 nM T58992 C1VB4E 10343492 EC50 = 135 nM T58992 C3P0LR 10345440 Ki = 56 nM T58992 C4BJ3Y 10346220 IC50 = 1.2 nM T58992 C15SJH 10346615 Ki = 573 nM T58992 CJXM25 10347927 Ki = 1.5 nM T58992 C8ZQB3 10350630 IC50 = 50 nM T58992 CPO17B 10351514 Ki = 2.1 nM T58992 CM6N1T 10358054 Ki > 10000 nM T58992 CPN1F0 10365429 Ki = 10.9 nM T58992 CCPH78 10366385 IC50 = 1700 nM T58992 C0ZF8R 10366960 IC50 = 120 nM T58992 C8VCR7 10374265 IC50 = 730 nM T58992 C7GK4U 10378392 Ki > 10000 nM T58992 CAYF18 10385808 Ki > 2000 nM T58992 CYD30U 10387038 Ki = 6.48 nM T58992 CX2EG6 10388274 IC50 = 8 nM T58992 C95EWP 10395965 Ki > 5000 nM T58992 CWK4O1 10406239 Ki = 4.9 nM T58992 CTA8Q0 10407144 Ki = 1492 nM T58992 CX6ZH1 10408431 IC50 = 264 nM T58992 CN5TB6 10408752 Ki = 275 nM T58992 CYWF17 10412617 IC50 = 4.9 nM T58992 CZ8UP5 10414887 IC50 = 3.2 nM T58992 CRN23P 10415050 Ki = 21.9 nM T58992 CUJL35 10415290 IC50 = 11.4 nM T58992 C6LBC5 10415925 Ki = 0.93 nM T58992 CD2P5F 10416962 Ki = 15 nM T58992 C7BVJ1 10428991 Ki = 200 nM T58992 C1U6NG 10430432 Ki = 93.9 nM T58992 CYHC38 10430819 Ki = 2137.96 nM T58992 C5G7NZ 10431410 Ki = 48.6 nM T58992 CQH92Z 10433421 Ki = 0.4 nM T58992 CON12X 10435156 EC50 = 0.95 nM T58992 CU51WV 10440134 Ki = 5.1 nM T58992 CQ4M0D 10443502 Ki = 5216 nM T58992 CS6E1O 10448420 Ki = 15 nM T58992 C7AQ0G 10449693 Ki = 72 nM T58992 CZ6I9V 10451761 IC50 > 10000 nM T58992 CV14CY 10452891 IC50 = 3 nM T58992 C7SOP4 10455862 IC50 = 17 nM T58992 C7DQ0Z 10455974 IC50 > 1000 nM T58992 C76HGO 10456060 Ki = 7.78 nM T58992 C5UG7N 10458677 Ki = 11 nM T58992 C2MY1U 10459444 IC50 = 1.3 nM T58992 CT39OH 10462262 IC50 = 2.4 nM T58992 C9T1SA 10463024 Ki > 100000 nM T58992 C3LT0F 10464136 IC50 = 17 nM T58992 C9C1JT 10473705 Ki = 54 nM T58992 CKMN08 10475466 Ki = 4680 nM T58992 CEF2O6 10478367 Ki > 10000 nM T58992 CT31DW 10479670 EC50 = 0.9 nM T58992 CPN21H 10481516 IC50 = 0.8 nM T58992 CE2LD8 10486131 Ki = 8.5 nM T58992 CS1L3N 10492792 IC50 = 1294 nM T58992 CWFU85 10496165 IC50 = 60.4 nM T58992 CKZ0V5 10498207 IC50 > 10000 nM T58992 CP72JI 10499145 IC50 = 15 nM T58992 C1DI7F 10500922 Ki = 1800 nM T58992 CGCP09 10501573 IC50 = 28.6 nM T58992 CQSG29 10508419 Ki = 0.5 nM T58992 CISG06 10508427 Ki = 6.81 nM T58992 CJ2BC7 10525105 EC50 = 18 nM T58992 CDGM01 10525171 EC50 = 54.6 nM T58992 C8FB2A 10527816 Ki > 1000 nM T58992 CT9U8L 10529438 Ki = 1.24 nM T58992 CU1AT8 10533341 Ki = 1.84 nM T58992 CNU8X2 10542105 Ki = 5700 nM T58992 C78MTF 10546451 Ki = 1500 nM T58992 C41JWE 10546813 EC50 = 303 nM T58992 CDK8W2 10548749 Ki = 480 nM T58992 CJ1TU0 10549849 IC50 = 2.09 nM T58992 CKP6E2 10550601 IC50 = 35.5 nM T58992 C71YXH 10553426 Ki = 4.93 nM T58992 CN4H7Z 10557001 Ki = 8.1 nM T58992 CKT1L0 10569964 IC50 = 11.3 nM T58992 C8E1UH 10570940 IC50 = 0.74 nM T58992 CLU72B 10572649 IC50 = 1.1 nM T58992 C54EOA 10572810 Ki = 1410 nM T58992 CD9JB5 10574643 Ki = 415 nM T58992 C28WNJ 10574908 Ki > 1000 nM T58992 C95XNB 10576543 IC50 = 13 nM T58992 C5Q4DU 10580071 Ki = 11 nM T58992 C79AIC 10592239 IC50 = 420 nM T58992 CQ74CO 10593778 Ki = 710 nM T58992 CT60BQ 10594839 IC50 = 27 nM T58992 CY6D1C 10596575 EC50 = 10.6 nM T58992 C2FL8C 10598391 EC50 = 10.4 nM T58992 C2CF1X 10598392 EC50 = 273 nM T58992 C71RMT 10599027 Ki = 1000 nM T58992 CHV5D1 10601891 Ki = 510 nM T58992 C6N5DI 10613803 IC50 = 509 nM T58992 CS84IW 10618605 Ki = 530 nM T58992 CK96NW 10618862 IC50 = 8.42 nM T58992 C62MNC 10620493 IC50 = 8 nM T58992 CIM8S1 10620902 EC50 = 0.9 nM T58992 CLC8U0 10628001 Ki = 0.66 nM T58992 CL14AV 10635842 Ki = 16 nM T58992 CA57UO 10636137 Ki > 5000 nM T58992 CBT4E1 10641623 IC50 = 100 nM T58992 CCV14H 10642101 IC50 = 98.4 nM T58992 C3CHZ0 10642670 IC50 = 1.04 nM T58992 C4XYH5 10644815 EC50 = 6.86 nM T58992 C9MY4Z 10644816 IC50 = 61.6 nM T58992 C8ZU7I 10644995 IC50 = 35.3 nM T58992 CF36MK 10645976 Ki = 494 nM T58992 CPC52U 10646744 Ki = 285 nM T58992 C10KTE 10646745 Ki = 240 nM T58992 CH32JY 10648307 IC50 = 7.5 nM T58992 C06MRN 10651237 Ki = 21.4 nM T58992 CA7Y6F 10651238 Ki = 61.1 nM T58992 CC4DN0 10651452 Ki = 19.9 nM T58992 CF0P6S 10662763 IC50 = 406 nM T58992 CC7MV8 10664865 IC50 = 100 nM T58992 C25PER 10664954 Ki = 1 nM T58992 CFC5R6 10668838 EC50 = 42.3 nM T58992 CP5L6A 10675111 Ki = 13.7 nM T58992 COQ80X 10675721 Ki = 74 nM T58992 CS8Y0V 10675722 Ki = 1.6 nM T58992 CY5BX7 10675737 Ki = 474 nM T58992 C84IHX 10676537 Ki = 9.5 nM T58992 CW92NR 10676779 Ki = 0.898 nM T58992 C64AHZ 10680393 Ki > 100000 nM T58992 CA0M1N 10690216 EC50 = 211 nM T58992 CBA6P3 10691980 IC50 > 2000 nM T58992 CGPT20 10692042 IC50 = 2.09 nM T58992 CVS40T 10695990 IC50 = 10.2 nM T58992 CHC1I4 10697286 Ki = 146 nM T58992 C3IWH5 10699409 Ki = 4.1 nM T58992 CAWZ71 10699417 Ki = 0.53 nM T58992 C1SIJ9 10706296 Ki > 10000 nM T58992 C5U4ZP 10713071 IC50 = 91.6 nM T58992 C8XB3K 10714523 Ki = 460 nM T58992 C2W9PN 10714960 IC50 = 4.17 nM T58992 CUAC76 10718278 Ki = 8.37 nM T58992 C8D2PI 10718445 Ki > 1000 nM T58992 C3E4PH 10718848 IC50 = 38 nM T58992 C82YCA 10719414 IC50 = 5 nM T58992 CV8K3J 10720494 Ki = 2.1 nM T58992 CAKS63 10722490 Ki = 34.9 nM T58992 CS84ZB 10722878 Ki = 2.91 nM T58992 C2VO1N 10735696 IC50 = 555 nM T58992 CS82CN 10739828 EC50 = 50 nM T58992 CAT04G 10741016 IC50 = 736 nM T58992 C8RW7M 10742582 Ki = 1.8 nM T58992 CF61KY 10742765 Ki = 8.22 nM T58992 CH17UA 10746795 Ki = 1.68 nM T58992 COW79X 10747714 Ki = 9.9 nM T58992 C4HD8E 10748690 IC50 = 820 nM T58992 C3CZ6L 10748691 IC50 = 65 nM T58992 C2J6UN 10756234 IC50 = 1045 nM T58992 CER5N6 10757499 Ki = 1600 nM T58992 C4BJ9L 10760345 IC50 = 8.77 nM T58992 CR4H2D 10760626 IC50 = 2.85 nM T58992 C0PT3I 10762996 EC50 = 44.9 nM T58992 CN05WO 10763594 Ki = 1380 nM T58992 CQ8EK9 10770328 Ki = 7.83 nM T58992 CIT9X3 10771171 Ki = 3478 nM T58992 CS1CE2 10771425 Ki = 7.8 nM T58992 CDJP34 10783436 IC50 > 10000 nM T58992 CK6J7P 10784079 IC50 = 2230 nM T58992 CB0JQ9 10785784 IC50 = 187 nM T58992 C54YIB 10786358 IC50 = 19.3 nM T58992 CSXE56 10787424 IC50 = 6.53 nM T58992 CE03JT 10788324 IC50 = 18 nM T58992 CZ58NT 10796106 Ki = 96.2 nM T58992 C74ONE 10804905 IC50 = 307 nM T58992 CU4WG6 10805007 Ki = 150 nM T58992 C2O0HR 10808721 IC50 = 2.57 nM T58992 C9G7LT 10809678 EC50 = 5.9 nM T58992 C3ZT7Y 10810430 Ki = 21.8 nM T58992 C0ZO7T 10811744 Ki = 22.1 nM T58992 CF0Q9U 10817984 Ki = 543 nM T58992 C2WNY5 10818843 Ki = 10.3 nM T58992 C0ZOE8 10818935 Ki = 9.7 nM T58992 C6BDP0 10827784 IC50 = 410 nM T58992 CS3Y4G 10832076 IC50 = 1900 nM T58992 CMVI50 10832445 Ki = 620 nM T58992 C9WI5X 10833535 IC50 = 2.04 nM T58992 C98NUA 10834101 IC50 = 37.89 nM T58992 CPG23C 10836379 Ki = 587 nM T58992 C4IT2B 10837001 Ki = 313 nM T58992 C8S5VW 10837156 IC50 = 26.6 nM T58992 CN0Z1M 10841295 Ki = 69 nM T58992 C1ZH8M 10841482 Ki = 37.7 nM T58992 CC8Z4K 10843252 Ki = 18 nM T58992 CB0I9F 10843787 IC50 = 140 nM T58992 C51ZGM 10843788 IC50 = 1050 nM T58992 C5Z9QW 10850629 Ki = 2400 nM T58992 C21TPE 10851779 Ki > 10000 nM T58992 C8K6UA 10853147 IC50 = 250 nM T58992 C13TAB 10853383 IC50 = 175 nM T58992 CFP68N 10872951 IC50 = 0.79 nM T58992 C7PR6B 10874095 EC50 = 0.65 nM T58992 C4ARK1 10883642 IC50 > 10000 nM T58992 C0H1TJ 10884365 IC50 > 10000 nM T58992 C9Y8OS 10884964 IC50 = 0.24 nM T58992 CB2QL0 10885771 IC50 > 10000 nM T58992 CR2D0K 10893581 IC50 = 4.9 nM T58992 CE6NR5 10893607 IC50 = 2 nM T58992 C0LM2D 10893958 IC50 = 5458 nM T58992 CF61NU 10895676 IC50 > 10000 nM T58992 CF3MG7 10897696 Ki = 40 nM T58992 CWJL70 10905740 IC50 = 620 nM T58992 CX65PW 10907460 IC50 = 8570 nM T58992 CRV83B 10907487 Ki = 1 nM T58992 CQ62UO 10918307 IC50 = 1765 nM T58992 CR21HO 10927114 Ki = 30902.95 nM T58992 CT79NZ 10927276 IC50 > 10000 nM T58992 C4TSV6 10927662 Ki = 1023.29 nM T58992 C1TSN4 10928037 Ki = 933.25 nM T58992 CTN91R 10929002 IC50 > 10000 nM T58992 C9M2JE 10929207 IC50 > 10000 nM T58992 C6G1ME 10930407 Ki = 21 nM T58992 CT5UO7 10937810 Ki = 1778.28 nM T58992 CU09AV 10937901 IC50 = 37.4 nM T58992 CM0OS2 10939174 IC50 > 10000 nM T58992 C6WQ3H 10939958 IC50 > 10000 nM T58992 CS42VZ 10941213 Ki = 99 nM T58992 CN7XS4 10948527 IC50 = 1190 nM T58992 CSLT97 10949380 IC50 = 117 nM T58992 CCUE70 10950205 IC50 > 10000 nM T58992 C9FYG3 10950562 Ki = 218.78 nM T58992 C48NDC 10950714 IC50 > 10000 nM T58992 CKR58N 10951763 Ki = 175 nM T58992 CHK23I 10961428 Ki = 1071.52 nM T58992 C2HP7F 10981761 IC50 = 4120 nM T58992 C32ZYJ 10982772 EC50 = 2.8 nM T58992 CMY56Q 10985930 Ki = 16200 nM T58992 CSZ6R2 10985963 Ki > 100000 nM T58992 C96ULE 10992239 IC50 = 1.3 nM T58992 CD5V9L 10992895 IC50 = 9.9 nM T58992 C91NTI 11003763 IC50 = 0.98 nM T58992 CJ6C9K 11003971 IC50 > 10000 nM T58992 C8Q6YE 11004121 Ki = 371.54 nM T58992 CJC9K4 11005810 IC50 = 5770 nM T58992 C3V7LT 11014751 Ki = 891.25 nM T58992 C8CP6J 11016127 IC50 = 0.22 nM T58992 C0VKL9 11016305 Ki = 118 nM T58992 C3WE6J 11024236 IC50 = 1.7 nM T58992 CC45BL 11025925 IC50 > 10000 nM T58992 CB7N1P 11035765 IC50 = 3330 nM T58992 CUI3F2 11046929 IC50 = 1410 nM T58992 C6EBF3 11048769 IC50 > 10000 nM T58992 C57NRV 11051174 Ki = 14100 nM T58992 CL8Z9G 11058283 Ki > 10000 nM T58992 CFJG64 11059058 IC50 = 2530 nM T58992 CL9Y8H 11059305 IC50 = 5640 nM T58992 C2ASJ3 11070421 Ki = 83.6 nM T58992 CWAB48 11071778 Ki = 0.63 nM T58992 C5ZP8L 11082539 Ki = 18600 nM T58992 CS4BM0 11090195 IC50 = 1.1 nM T58992 CR0TL9 11091522 IC50 = 0.33 nM T58992 CA68BR 11091606 Ki = 1090 nM T58992 CO08EV 11091686 IC50 > 10000 nM T58992 C6HIQ0 11092200 IC50 = 7130 nM T58992 C7WB6K 11094406 Ki = 13200 nM T58992 CONE61 11104644 Ki = 12600 nM T58992 CF0SV1 11112699 IC50 = 0.99 nM T58992 C7DE0U 11113605 IC50 = 9380 nM T58992 CJ25OQ 11122114 IC50 > 10000 nM T58992 C3CGB7 11123013 IC50 = 0.79 nM T58992 CM9P2I 11123816 EC50 = 0.87 nM T58992 CDU0E5 11123873 Ki = 2951.21 nM T58992 C6P5EL 11129476 Ki = 9750 nM T58992 C9WXY1 11132954 Ki > 10000 nM T58992 CN8UZ0 11136722 Ki = 15100 nM T58992 C04HTO 11139094 IC50 > 10000 nM T58992 CIL4S3 11140284 Ki = 1050 nM T58992 CU6PV0 11143820 IC50 = 138 nM T58992 CP96WD 11145858 IC50 = 0.29 nM T58992 CPW06I 11146107 Ki = 2 nM T58992 C10FGZ 11149261 Ki = 3830 nM T58992 CEW8Z0 11149937 Ki = 1200 nM T58992 C8W9RO 11150306 Ki = 13 nM T58992 CS90VC 11153600 Ki > 10000 nM T58992 C9FCD2 11153683 Ki > 1000 nM T58992 C4NAJ5 11154544 Ki = 170 nM T58992 CE6N5V 11157443 Ki = 23.91 nM T58992 C67ZFK 11158498 Ki = 400 nM T58992 CJO8S0 11163232 Ki = 940 nM T58992 CF7QE8 11163411 Ki > 10000 nM T58992 C6A0JS 11166820 Ki = 37 nM T58992 C26PQJ 11167140 Ki > 10000 nM T58992 C0DO8C 11175032 Ki > 10000 nM T58992 C16TCJ 11180190 Ki > 1000 nM T58992 CPQ6A8 11180584 Ki = 15.48 nM T58992 CM9TV6 11181676 Ki = 80 nM T58992 CLE18Z 11184156 Ki = 2220 nM T58992 CAKZ38 11184946 IC50 > 10000 nM T58992 CPOD70 11186271 Ki = 595 nM T58992 CM6Q2S 11186913 Ki = 93 nM T58992 CAZ30T 11188794 Ki = 79 nM T58992 C90HXY 11190061 Ki = 3.9 nM T58992 CMRJ71 11191431 Ki = 230 nM T58992 CJL1R5 11198030 Ki = 591 nM T58992 CE6HS7 11200189 Ki = 2.7 nM T58992 CIG2Q9 11201660 Ki = 167 nM T58992 CGL3W7 11204993 Ki = 32 nM T58992 CSQ73J 11209418 Ki = 1900 nM T58992 CD3J8L 11209549 Ki = 600 nM T58992 CIAE47 11211122 Ki = 2.5 nM T58992 CK42LP 11213149 EC50 = 1.4 nM T58992 CBV6X8 11213578 Ki = 1.56 nM T58992 CZ4US0 11215747 Ki = 19.18 nM T58992 CK8VG1 11220535 Ki = 472 nM T58992 CN8LV4 11235302 EC50 = 37 nM T58992 C7LD4V 11238343 Ki = 26.81 nM T58992 CA5T0Z 11238737 Ki = 85.05 nM T58992 C7DJ3L 11239327 Ki = 3.8 nM T58992 C8BO9A 11246669 Ki = 1.2 nM T58992 C6V7LK 11259665 Ki = 0.152 nM T58992 C1O5ZD 11262815 Ki = 21 nM T58992 CF4LV5 11264459 Ki = 4010 nM T58992 C3D7SY 11266864 Ki > 10000 nM T58992 CN12PC 11268925 Ki = 1800 nM T58992 CRZ3V0 11269310 Ki = 1.8 nM T58992 C9LFY6 11269707 Ki = 0.6 nM T58992 CD19XU 11270347 Ki = 1125 nM T58992 CMI48S 11271318 Ki > 10000 nM T58992 CK90ZB 11271551 Ki = 0.24 nM T58992 C3G6PC 11273472 Ki = 95.82 nM T58992 CPBZ36 11274537 Ki > 5000 nM T58992 CHYM79 11279188 Ki = 4 nM T58992 C5WYA8 11280721 Ki = 7.4 nM T58992 CGOV28 11282704 IC50 = 74 nM T58992 CP27SY 11283686 IC50 = 0.25 nM T58992 CTX1Y0 11292839 IC50 = 920 nM T58992 CQ0FP3 11292970 Ki = 10000 nM T58992 CFR9X1 11302996 Ki > 10000 nM T58992 C59MLX 11305998 Ki = 6460 nM T58992 CR4TD3 11307039 Ki = 600 nM T58992 CAWZ12 11308699 Ki = 920 nM T58992 CF60BC 11308721 Ki = 24 nM T58992 CAOJ05 11311787 Ki = 672 nM T58992 C8P5AT 11314197 Ki > 4000 nM T58992 C4FRH7 11315651 Ki > 400 nM T58992 C9A1PL 11318909 Ki = 8.52 nM T58992 CR85OX 11319221 Ki = 15.04 nM T58992 CMK6Q8 11322246 Ki > 10000 nM T58992 C5DBK1 11326750 IC50 > 10000 nM T58992 CI94VH 11327829 Ki = 380 nM T58992 C9D4TI 11330655 Ki = 41.86 nM T58992 CI4SY0 11333521 Ki = 2430 nM T58992 CIS8B5 11334123 Ki = 2090 nM T58992 COM5A1 11335412 Ki = 2300 nM T58992 C7O0ER 11337925 Ki = 1.6 nM T58992 CIG49E 11339827 Ki = 5.9 nM T58992 C4C0OE 11341622 Ki = 6470 nM T58992 C10YKF 11351067 Ki > 10000 nM T58992 C13ERF 11351769 Ki = 1.1 nM T58992 CJ9P1G 11352435 Ki = 1500 nM T58992 C4CFD0 11358487 Ki = 5770 nM T58992 CB5F8T 11359173 Ki = 74 nM T58992 C5H2OX 11359253 Ki = 410 nM T58992 CME1I6 11359624 Ki > 1000 nM T58992 C7EUO6 11361718 EC50 = 542 nM T58992 CLT47S 11364225 Ki = 44 nM T58992 C73GIN 11365113 Ki = 370 nM T58992 CA19LC 11373068 Ki = 3.7 nM T58992 C9HGE1 11374952 Ki > 10000 nM T58992 C1WBH7 11375776 EC50 = 1.9 nM T58992 CZS3E9 11376776 Ki = 7.24 nM T58992 C2E8MJ 11382472 Ki = 5.6 nM T58992 CH50TV 11388486 Ki = 16 nM T58992 C5OIU1 11391288 Ki = 601 nM T58992 CR9V8F 11391721 Ki = 2720 nM T58992 C76WKY 11392900 Ki > 10000 nM T58992 CV5PY7 11394342 Ki = 9.7 nM T58992 CCK72R 11402990 Ki = 2500 nM T58992 C5QBV4 11404339 Ki = 690 nM T58992 CJL06W 11404566 Ki = 1 nM T58992 C29SLF 11405480 Ki = 50 nM T58992 CQE92F 11406708 Ki = 0.69 nM T58992 C6S9EV 11416117 Ki = 1100 nM T58992 C6BE9Q 11417954 Ki = 0.84 nM T58992 CBGR89 11419799 Ki > 10000 nM T58992 C4S8GN 11421830 Ki = 17.58 nM T58992 CML2H3 11428837 Ki = 1.8 nM T58992 CS9G3B 11430490 Ki = 2.3 nM T58992 CY5Z6D 11434336 Ki = 82 nM T58992 CSZ2F1 11440849 EC50 = 14 nM T58992 C9R7AI 11444917 Ki = 18.06 nM T58992 CN40IB 11449538 Ki > 10000 nM T58992 C7Y2CR 11451042 Ki = 800 nM T58992 CY7HT3 11452117 Ki = 3.5 nM T58992 C3M4ZJ 11455086 Ki = 15 nM T58992 C7UDE8 11461888 Ki > 10000 nM T58992 CMU9K5 11464846 Ki > 400 nM T58992 CMV04H 11470285 Ki = 5830 nM T58992 CO95HP 11474838 Ki = 0.43 nM T58992 C3T5SC 11479033 Ki = 6.73 nM T58992 C3BA5F 11480038 Ki > 5000 nM T58992 C4XU0O 11486901 Ki > 10000 nM T58992 C1LJ5U 11487063 Ki > 10000 nM T58992 C5UR1M 11487946 Ki = 7823 nM T58992 CA4PM8 11496383 EC50 = 380 nM T58992 CX6Q0I 11497325 Ki = 9330 nM T58992 CQP65V 11503501 Ki = 0.62 nM T58992 C5YIE4 11510112 Ki = 990 nM T58992 C41MEV 11511090 IC50 > 10000 nM T58992 C2E7LB 11511362 Ki = 510 nM T58992 C5LA3M 11521945 Ki = 2400 nM T58992 CQ30PM 11525624 IC50 > 10000 nM T58992 C49XZQ 11526334 Ki = 7620 nM T58992 CB1K8W 11533999 Ki = 3720 nM T58992 CF86WQ 11537712 Ki = 150 nM T58992 CB2U5X 11540292 EC50 = 380 nM T58992 C07WHY 11541833 EC50 > 1000 nM T58992 C8TZ9G 11544654 IC50 > 10000 nM T58992 COF4K0 11544824 Ki = 460 nM T58992 CHI36N 11547640 Ki = 4240 nM T58992 CHI47M 11555262 Ki > 10000 nM T58992 CT95KX 11555338 IC50 = 5.012 nM T58992 C2ZNA4 11558993 Ki = 480 nM T58992 C97WYH 11559278 Ki = 80 nM T58992 CVI52T 11561040 Ki > 10000 nM T58992 CO02FI 11562377 EC50 = 380 nM T58992 C3E4LV 11562400 Ki = 1380 nM T58992 CVA8L6 11583016 IC50 > 10000 nM T58992 C3PX0F 11584092 Ki > 10000 nM T58992 CO0N2L 11591805 Ki = 3.7 nM T58992 CZA48L 11591838 Ki > 10000 nM T58992 C9GPQ8 11595485 Ki = 2600 nM T58992 C1WBQ5 11597677 IC50 > 10000 nM T58992 CE4ZV5 11602862 Ki = 130 nM T58992 C8RKH0 11619553 IC50 > 10000 nM T58992 CSYE45 11619680 EC50 = 380 nM T58992 CM8NO4 11628123 Ki > 10000 nM T58992 C4ZD1X 11633324 IC50 > 10000 nM T58992 CZ05OM 11641014 Ki = 510 nM T58992 C2USB1 11655841 Ki = 3970 nM T58992 CC1EZ6 11657075 Ki > 10000 nM T58992 CQML27 11660069 Ki = 1050 nM T58992 CS91JQ 11666402 Ki = 2100 nM T58992 CXO5K2 11667199 Ki > 10000 nM T58992 C9XD2T 11677662 Ki = 18 nM T58992 CW7QD2 11698381 EC50 = 380 nM T58992 C19DJE 11698420 EC50 = 380 nM T58992 C79XSW 11705263 Ki = 4030 nM T58992 C4ULQ7 11710187 IC50 > 10000 nM T58992 C4PXV7 11712760 EC50 = 380 nM T58992 CUG57V 11713930 Ki > 10000 nM T58992 C8A2CG 11714559 Ki = 1.8 nM T58992 CC4SF3 11717551 Ki = 900 nM T58992 COL07J 11728653 IC50 = 0.97 nM T58992 C7FSD3 11729952 IC50 = 0.41 nM T58992 C7PVL8 11730467 IC50 = 3710 nM T58992 CV3OY7 11733074 IC50 > 10000 nM T58992 CCN8E9 11742939 IC50 = 1.15 nM T58992 CPG15O 11743399 IC50 > 1000 nM T58992 CE0D1U 11743914 Ki = 9385 nM T58992 CS60CA 11750461 EC50 = 85 nM T58992 CBH0Y7 11753736 Ki = 5.05 nM T58992 CF6M2I 11755589 Ki = 105.7 nM T58992 CFRY36 11757207 Ki = 777 nM T58992 C3F5DX 11761059 IC50 = 1040 nM T58992 CED7I5 11761926 Ki = 389.05 nM T58992 CEI7T9 11771732 Ki = 260 nM T58992 CC61WX 11773726 Ki = 1.05 nM T58992 CX27WK 11779453 Ki = 7.6 nM T58992 CJ7L9W 11784235 IC50 = 3.2 nM T58992 C1K0JF 11786990 Ki = 11.7 nM T58992 C7TLS3 11793476 EC50 = 53.3 nM T58992 CJD95Z 11794240 IC50 = 24.8 nM T58992 C1LJM6 11794241 IC50 = 8.13 nM T58992 CG9HW8 11795019 Ki = 450 nM T58992 C5C8NP 11795327 Ki > 300 nM T58992 CW69HO 11795406 IC50 = 132 nM T58992 C60RKP 11796211 IC50 = 2.31 nM T58992 C80ZJV 11797669 Ki = 2.94 nM T58992 C4SCZ1 11797670 Ki = 34.5 nM T58992 CJ10CQ 11803174 Ki = 7.1 nM T58992 COSJ52 11811375 IC50 = 1.1 nM T58992 CN9M8E 11811722 IC50 = 1840 nM T58992 CXY38K 11812228 IC50 > 10000 nM T58992 CJ6AL3 11818885 IC50 = 1740 nM T58992 C8UE5W 11826819 Ki = 912.01 nM T58992 CC65TG 11827053 EC50 = 1.7 nM T58992 CS7W2V 11848793 Ki = 2326 nM T58992 C65TDJ 11849246 IC50 = 248 nM T58992 CHV25L 11849247 Ki = 2.3 nM T58992 CQ6P3Y 11849249 Ki = 1.3 nM T58992 CIKN38 11849282 Ki = 1.25 nM T58992 CR47EN 11849283 Ki = 2.9 nM T58992 C7SI8L 11849284 Ki = 0.42 nM T58992 CP8QH4 11849285 Ki = 0.11 nM T58992 C7D2TB 11849360 Ki = 1 nM T58992 CK2RQ0 11849361 Ki = 0.58 nM T58992 CD39RT 11849364 Ki = 7.2 nM T58992 C63YAV 11849365 IC50 = 21.2 nM T58992 CXLW54 11948707 Ki > 10000 nM T58992 CS0MC4 11950654 EC50 = 7500 nM T58992 CEVH83 12041054 Ki = 10 nM T58992 CJP1W3 12041055 Ki = 2.38 nM T58992 C5RD1S 12041056 Ki = 0.7 nM T58992 CQ1B6S 12048050 Ki = 2780 nM T58992 C03DLA 12093958 Ki = 148 nM T58992 CYCF29 12103026 IC50 > 10000 nM T58992 CY7X8O 12112720 Ki > 10000 nM T58992 CT9KA1 12114808 Ki > 5200 nM T58992 CBK43E 12114809 Ki > 5200 nM T58992 C6IT0O 12191611 Ki > 10000 nM T58992 CYBD81 12191612 Ki = 44 nM T58992 CS5IZ8 12371110 Ki = 449 nM T58992 CSY9N8 12371111 Ki = 7000 nM T58992 CQI8H1 12802420 IC50 = 230 nM T58992 CXF1M5 12988885 Ki = 35 nM T58992 C8K6DU 12994684 Ki = 2.6 nM T58992 CAR89Y 12994686 Ki = 12 nM T58992 CPV4D2 13062443 Ki = 1640 nM T58992 CZ0AH1 13062446 Ki = 17500 nM T58992 CVO34T 13559317 Ki = 46.2 nM T58992 CNJ1Q6 13559325 Ki = 8.8 nM T58992 C06ADH 13599612 Ki > 10000 nM T58992 C74GFU 14548197 IC50 > 10000 nM T58992 CO9LG8 14548199 IC50 > 10000 nM T58992 CWC40I 14548201 IC50 > 10000 nM T58992 C6ZGM1 14548203 IC50 > 10000 nM T58992 C1OBG5 14548205 IC50 > 10000 nM T58992 C07XRE 14548207 IC50 > 10000 nM T58992 C6NAX7 14548209 IC50 > 10000 nM T58992 C5PEH8 14548211 IC50 > 10000 nM T58992 CZJ64M 14548213 IC50 > 10000 nM T58992 C81RSB 14548215 IC50 > 10000 nM T58992 C4RAE8 14548217 IC50 > 10000 nM T58992 CUK2G3 14548219 IC50 > 10000 nM T58992 CHRI24 14548221 IC50 = 2300 nM T58992 C1N7OD 14548223 IC50 = 9000 nM T58992 CG9L2K 14548225 IC50 > 10000 nM T58992 CP0K1I 14548227 IC50 = 5800 nM T58992 C71ALD 14548229 IC50 > 10000 nM T58992 CKCB61 14548236 IC50 = 6300 nM T58992 CGQK84 14548238 IC50 > 10000 nM T58992 C9C5TY 14570180 Ki = 4270 nM T58992 C0UX9N 14570184 Ki = 2690 nM T58992 C9Y6MU 14679812 Ki = 1.7 nM T58992 C7M2XS 14726012 Ki = 113 nM T58992 C3XU4Q 14810985 Ki > 10000 nM T58992 C0KRX7 14810989 Ki > 10000 nM T58992 CJCX20 14810996 Ki > 10000 nM T58992 CY5Q3K 14845809 Ki = 38 nM T58992 CVF09U 14879862 IC50 = 809 nM T58992 CQ9O3D 14879863 IC50 = 1701 nM T58992 CM5OY7 15130837 Ki = 1850 nM T58992 CL9E5Q 15130838 Ki = 3070 nM T58992 C9UIM1 15160017 IC50 = 18.6 nM T58992 CRI0E5 15177772 Ki > 100000 nM T58992 CKU83M 15177773 Ki = 9510 nM T58992 CJNP94 15177774 Ki = 12300 nM T58992 CF27TQ 15384274 Ki = 2.7 nM T58992 CUND10 15407235 IC50 = 4969 nM T58992 CAW1M2 15512228 Ki < 501.19 nM T58992 C30CHU 15512229 Ki = 100 nM T58992 CX6H8V 15512234 Ki = 158.49 nM T58992 CC5X0L 15512235 Ki < 501.19 nM T58992 C53KRM 15512237 Ki = 158.49 nM T58992 CLA5K8 15512238 Ki < 501.19 nM T58992 CSX74V 15512240 Ki < 501.19 nM T58992 CET25R 15512241 Ki < 501.19 nM T58992 C7CNY1 15512243 Ki < 501.19 nM T58992 CZA4J8 15541261 Ki = 37890 nM T58992 CRM01L 15548354 Ki = 63.2 nM T58992 C1DB3A 15548355 Ki = 451 nM T58992 CCN3D0 15659189 Ki = 1.1 nM T58992 C3YA2J 15659190 Ki = 3.27 nM T58992 CMB31A 15659191 Ki = 2.89 nM T58992 CM7TD0 15659192 Ki = 0.98 nM T58992 C7K9ZV 15659193 Ki = 5.38 nM T58992 CWU53Z 15659194 Ki = 36.7 nM T58992 C20OCE 15659195 Ki = 25.6 nM T58992 CPC71O 15659196 Ki = 9.29 nM T58992 C0XN5S 15659197 Ki = 1.66 nM T58992 CA5F8L 15663405 IC50 = 12 nM T58992 CSR70J 15663406 IC50 = 13 nM T58992 C2EZL9 15663417 IC50 = 7.2 nM T58992 CL9O5E 15663418 IC50 = 7.7 nM T58992 CLJ7K9 15663419 IC50 = 9.1 nM T58992 C4T3ZN 15663420 IC50 = 19 nM T58992 CZD82L 15689703 Ki = 10100 nM T58992 C37CJK 15689709 Ki = 22700 nM T58992 CQL2N9 15689712 Ki > 10000 nM T58992 CPOR80 15689718 Ki = 8430 nM T58992 CBZW58 15697369 Ki > 1000 nM T58992 CGOY52 15697372 Ki = 153 nM T58992 CUZV36 15697375 Ki > 1000 nM T58992 C1RM9L 15697378 Ki > 1000 nM T58992 CYR35U 15697379 Ki > 1000 nM T58992 CA7FK6 15697380 Ki > 1000 nM T58992 C4NQ5C 15819291 Ki = 4.9 nM T58992 C9TYD1 15923664 Ki = 24 nM T58992 C75LOT 15934554 Ki = 1500 nM T58992 C6DW5M 15982528 IC50 > 10000 nM T58992 C7Z8OD 15982529 IC50 > 10000 nM T58992 CHO67K 15982530 IC50 > 10000 nM T58992 CV1G7O 15982660 IC50 > 10000 nM T58992 CG3L8Z 15982661 IC50 > 10000 nM T58992 CN64AP 15982791 IC50 > 10000 nM T58992 CJ6W1T 15982933 IC50 > 10000 nM T58992 CG96OQ 15983067 IC50 > 10000 nM T58992 CV3TQ9 16006949 Ki = 0.74 nM T58992 CA5GL7 16007142 Ki > 5000 nM T58992 CK3QD9 16039356 Ki = 5250 nM T58992 CI8FE0 16046123 Ki = 0.99 nM T58992 C3XA7E 16048783 Ki = 12 nM T58992 CDV05T 16048784 Ki = 72 nM T58992 C3O4HX 16048863 Ki = 0.72 nM T58992 CPV60X 16048864 Ki = 0.71 nM T58992 CFZI17 16048866 Ki = 2.5 nM T58992 CNDV23 16048867 Ki = 3.5 nM T58992 C9SCH7 16048936 Ki = 150 nM T58992 C6A5UL 16048937 Ki = 24 nM T58992 C3PO9S 16048938 Ki = 0.9 nM T58992 CJ6LM3 16048939 Ki = 18 nM T58992 CUQ16Z 16048940 Ki = 18 nM T58992 CG71OP 16048941 Ki = 5.9 nM T58992 CP23YA 16049012 Ki = 21 nM T58992 CQK63V 16051935 IC50 = 242 nM T58992 C6LFA8 16059781 Ki = 1860 nM T58992 C7ZDK2 16082868 IC50 = 95 nM T58992 CRM3G1 16082874 IC50 = 0.42 nM T58992 CS8I2H 16082875 IC50 = 0.68 nM T58992 CEA34Z 16082876 IC50 = 0.39 nM T58992 CX6VJ0 16082877 IC50 = 0.4 nM T58992 CY7I6C 16082878 IC50 = 1.8 nM T58992 C4D7FJ 16082879 IC50 = 0.15 nM T58992 C7JA5T 16082880 IC50 = 0.48 nM T58992 CY4LT1 16082881 IC50 = 0.45 nM T58992 C2VO3C 16082882 IC50 = 16 nM T58992 CG64ZK 16082883 IC50 = 7.7 nM T58992 C2JR9P 16082884 IC50 = 0.45 nM T58992 C2B5OD 16082889 IC50 = 1.4 nM T58992 CCI10V 16082892 IC50 = 0.12 nM T58992 CP50WM 16082893 IC50 = 0.72 nM T58992 CG14FD 16082894 IC50 = 0.8 nM T58992 CJ4M6R 16082913 IC50 = 0.5 nM T58992 CSK23U 16083041 Ki = 0.24 nM T58992 CQR13T 16086545 IC50 = 75400 nM T58992 CR0S9Y 16087270 IC50 = 0.03 nM T58992 CSB90O 16087271 IC50 = 1.7 nM T58992 C75QOB 16087272 IC50 = 3.35 nM T58992 CP5B0A 16087273 IC50 = 1.17 nM T58992 CK8C3L 16087274 Ki = 1.51 nM T58992 CBW82T 16087275 IC50 = 0.76 nM T58992 CFZ95P 16087276 Ki = 242 nM T58992 C48WDR 16087277 IC50 = 79.9 nM T58992 C7V4ZB 16087278 Ki = 24.8 nM T58992 C8X5HT 16087279 Ki = 55.9 nM T58992 CE7G1T 16087280 Ki = 33.8 nM T58992 C4B1NT 16087283 IC50 = 0.02 nM T58992 CU1J5C 16087284 IC50 = 1.37 nM T58992 CU15KC 16087285 IC50 = 0.67 nM T58992 C30MPR 16087286 IC50 = 1.59 nM T58992 CITF65 16087287 IC50 = 1.66 nM T58992 CN5KV0 16087288 Ki = 104 nM T58992 C4FW9H 16087289 Ki = 94.9 nM T58992 C2OVH1 16087290 Ki = 51.9 nM T58992 C3S7GV 16094319 Ki = 190 nM T58992 CR71BM 16094320 Ki = 25 nM T58992 CV1P4O 16094322 Ki = 220 nM T58992 CZ4V9I 16094342 Ki = 900 nM T58992 CO8T5W 16094343 Ki = 31 nM T58992 C0I9GV 16094344 Ki = 2.1 nM T58992 C21JYZ 16094345 Ki = 280 nM T58992 CB4NE1 16094362 Ki = 1700 nM T58992 C3SZX8 16094366 Ki = 2900 nM T58992 C5RGW0 16094367 IC50 = 62 nM T58992 CB46JH 16094368 Ki = 510 nM T58992 CCLO14 16094369 Ki = 350 nM T58992 CUN6E1 16094370 Ki = 57 nM T58992 C9QI4H 16094371 Ki = 360 nM T58992 C90BWG 16094372 Ki = 420 nM T58992 CTY5V3 16094373 Ki = 300 nM T58992 C23KIF 16094374 Ki = 310 nM T58992 C48EXZ 16094375 Ki = 220 nM T58992 CL1A7O 16094383 Ki = 1100 nM T58992 CKS40Z 16094384 Ki = 840 nM T58992 CDG2M6 16094385 Ki = 1300 nM T58992 C5WZF1 16094386 Ki = 1500 nM T58992 CYP92H 16094387 Ki = 740 nM T58992 CGRX31 16094388 Ki = 260 nM T58992 CO4Z1K 16094389 Ki = 340 nM T58992 CH23IJ 16094390 Ki = 65 nM T58992 CS8L3K 16094394 Ki = 340 nM T58992 CX87TS 16094397 Ki = 1100 nM T58992 C4RIZ1 16094408 Ki = 660 nM T58992 C4D1UF 16094410 Ki = 410 nM T58992 CUA2L0 16094413 Ki = 71 nM T58992 C3AMW5 16094414 Ki = 140 nM T58992 C6J0YV 16094415 Ki = 960 nM T58992 CX4K0L 16094416 Ki = 540 nM T58992 CR7AS8 16094419 Ki = 960 nM T58992 CK98PS 16094420 Ki = 89 nM T58992 C9AJK7 16094421 IC50 = 580 nM T58992 C57IQS 16094423 Ki = 2500 nM T58992 CI2XK6 16094424 Ki = 60 nM T58992 C6GL2A 16094425 IC50 = 33 nM T58992 CO4M3A 16094426 IC50 = 28 nM T58992 C1JBM6 16094428 IC50 = 14 nM T58992 CMI74R 16094429 Ki = 140 nM T58992 CK7N1Y 16094430 Ki = 240 nM T58992 C3T9MH 16100406 Ki = 3.9 nM T58992 CH6F0V 16100408 Ki = 6.9 nM T58992 CI7FD0 16105558 EC50 > 1000 nM T58992 C7S6KX 16105562 EC50 > 1000 nM T58992 CW17YU 16224209 Ki = 1517 nM T58992 CZ18VL 16224211 Ki = 3.2 nM T58992 CSG27D 16224612 Ki = 3.5 nM T58992 CK5GY1 16224613 Ki = 0.58 nM T58992 CZ2IS9 16660294 Ki > 10000 nM T58992 C08RXS 16665915 Ki > 5000 nM T58992 CS9FW1 16665917 Ki > 5000 nM T58992 C1LX0I 16665918 Ki > 5000 nM T58992 CCF0J7 16720551 Ki = 1.5 nM T58992 C0ACW1 16720553 Ki = 0.35 nM T58992 CG6OD7 16720646 Ki = 0.17 nM T58992 CC4N5P 16720648 Ki = 13 nM T58992 CFI67Y 16720649 Ki = 4.2 nM T58992 C8GOL2 16720650 Ki = 1.1 nM T58992 CB9MZ5 16720745 EC50 = 0.16 nM T58992 CAY72B 16720746 Ki = 35 nM T58992 CO84NU 16720747 Ki = 8.7 nM T58992 CG62NU 16720749 EC50 = 0.17 nM T58992 C4U5XO 16730656 EC50 = 59 nM T58992 C8KRM1 16730814 EC50 = 27 nM T58992 C2CRF5 16730815 EC50 = 12 nM T58992 C8SOD5 16735664 Ki = 2.25 nM T58992 CG9WC1 16735704 EC50 = 16.6 nM T58992 C20SRH 16737292 Ki = 15 nM T58992 C9GZ7X 16737294 Ki = 36 nM T58992 C9MZD1 16737629 Ki = 5 nM T58992 C0EBA3 16737631 EC50 = 1.8 nM T58992 C23MPB 16737673 Ki = 2.8 nM T58992 C4ORI6 16739256 Ki = 11655 nM T58992 C1MFJ2 16747695 Ki = 518 nM T58992 C4P0RO 16747723 IC50 = 32100 nM T58992 C5UGV2 16748227 Ki > 10000 nM T58992 CO0XL6 16748228 Ki > 10000 nM T58992 CNEX42 16748229 Ki > 10000 nM T58992 CN4JB2 16748352 Ki > 10000 nM T58992 CJX60K 16748353 Ki > 10000 nM T58992 C5W1UD 16748354 Ki > 10000 nM T58992 C9ZD4O 16748355 Ki > 10000 nM T58992 C9TC3L 16748356 Ki > 10000 nM T58992 C68VNE 16748478 Ki > 10000 nM T58992 C6QMJ9 16756731 Ki = 4600 nM T58992 C4AEU1 16756734 Ki = 1570 nM T58992 C9D5RB 16756735 Ki = 720 nM T58992 C2BG6Z 16756840 Ki = 13 nM T58992 C0Q2OC 16756841 Ki = 2735 nM T58992 C6NF5U 16756953 Ki = 770 nM T58992 CS26LH 16757050 Ki = 90 nM T58992 CFS39T 16757147 Ki = 300 nM T58992 C7QJW9 17379334 Ki = 3 nM T58992 CJY27L 17798965 Ki = 163 nM T58992 C6IW7Z 17798971 Ki = 176 nM T58992 CIQ2R5 17798973 Ki = 710 nM T58992 CX91VE 17798974 Ki > 10000 nM T58992 CGB04N 17798976 Ki = 781 nM T58992 CYJ06B 17798978 Ki > 10000 nM T58992 CJNQ89 17925232 Ki = 2.9 nM T58992 C0H1TB 18545701 Ki = 4.5 nM T58992 C1Y9FT 18782352 Ki = 2650 nM T58992 CYUG80 18782376 Ki = 2511 nM T58992 C46DPT 18782378 Ki = 2266 nM T58992 C73DWV 18782384 Ki = 1906 nM T58992 C61OBX 19881394 Ki = 1315 nM T58992 C7T8JC 19958494 Ki > 10000 nM T58992 C6LI5E 19958507 Ki > 10000 nM T58992 C5BE7T 20345831 IC50 = 40 nM T58992 C3I8EH 20642899 Ki = 3500 nM T58992 C94FLX 20833183 IC50 = 12.1 nM T58992 CIOT38 20968607 IC50 > 32000 nM T58992 CP1HK3 21106890 Ki = 1369 nM T58992 C3T5HF 21509921 Ki > 10000 nM T58992 CBN84K 22065997 Ki > 10000 nM T58992 CS24KZ 22213385 Ki = 201 nM T58992 CHAI36 22272877 IC50 > 1000 nM T58992 C1W7MX 22522554 IC50 > 32000 nM T58992 C90UPB 22553442 IC50 > 32000 nM T58992 C1R5PV 22562132 Ki > 2000 nM T58992 CJ8OB0 22562135 Ki > 2000 nM T58992 C5YZ9U 22573205 Ki = 370 nM T58992 CKI1O3 22573217 Ki = 1000 nM T58992 CD4C5N 22729898 Ki = 0.9 nM T58992 CX3O6L 22729907 Ki = 1.9 nM T58992 C7OL1R 22729922 Ki = 11 nM T58992 CA28YU 22729923 Ki = 9 nM T58992 CG60MD 22816300 Ki = 241 nM T58992 CL7X2U 23383556 Ki = 867 nM T58992 COHN67 23383564 Ki = 606 nM T58992 CBW20U 23435898 IC50 = 1.56 nM T58992 C3HB1O 23519701 Ki = 9.8 nM T58992 C8ZD9W 23567095 Ki > 5000 nM T58992 C3K6HV 23594220 Ki = 63 nM T58992 CXC6E3 23594223 Ki = 83 nM T58992 CQ93SH 23594225 Ki = 167 nM T58992 CC5E7N 23594227 Ki = 513 nM T58992 CG3M5J 23594230 Ki = 107 nM T58992 C5L8ZA 23594232 Ki = 238 nM T58992 C08XMZ 23594241 Ki = 124 nM T58992 C0D5AC 23594243 Ki = 470 nM T58992 C4JGI8 23594247 Ki = 27 nM T58992 C2LIV7 23634920 Ki = 3.7 nM T58992 C2KP4M 23634921 Ki = 6.1 nM T58992 CI65DR 23635042 Ki = 7000 nM T58992 CW5QE4 23635163 Ki = 14 nM T58992 C9NLO3 23635166 Ki = 3.2 nM T58992 CXN07F 23661598 Ki = 2.3 nM T58992 C8TEB0 23723457 EC50 = 54 nM T58992 CO5YP3 23986637 Ki = 1.1 nM T58992 CB9MC8 24735827 Ki = 31935 nM T58992 C84JOU 24754997 Ki = 144.07 nM T58992 CPY62V 24762741 IC50 = 30900 nM T58992 CEF65A 24768357 Ki = 1.8 nM T58992 CN3AY8 24768358 Ki = 77 nM T58992 CH9E3R 24768397 Ki = 0.36 nM T58992 CWP85S 24776395 Ki > 10000 nM T58992 CVD48X 24776396 Ki > 10000 nM T58992 C3WDL8 24776397 Ki > 10000 nM T58992 CXL4R0 24776398 Ki > 10000 nM T58992 CR9I1S 24776399 Ki > 10000 nM T58992 CQDJ35 24776400 Ki > 10000 nM T58992 C6CX0Z 24776401 Ki > 10000 nM T58992 CJH18I 24776402 Ki > 10000 nM T58992 C27SGI 24776403 Ki > 10000 nM T58992 CV5IG2 24776404 Ki > 10000 nM T58992 CQ70IW 24776405 Ki > 10000 nM T58992 CQ2P5J 24776406 Ki > 10000 nM T58992 CYIV42 24776407 Ki > 10000 nM T58992 CWB06Z 24776408 Ki > 10000 nM T58992 C36WQO 24776409 Ki > 10000 nM T58992 CUP2C6 24776410 Ki > 10000 nM T58992 CC3W7E 24776411 Ki > 10000 nM T58992 C3N6GE 24776412 Ki > 10000 nM T58992 C2M6BR 24776413 Ki > 10000 nM T58992 CL2WB0 24800108 Ki > 667 nM T58992 CFIS62 24822296 Ki = 17.59 nM T58992 CB4S7U 24822297 Ki = 36.52 nM T58992 CC06ON 24822298 Ki = 25.29 nM T58992 C30GOT 24822299 Ki = 3.1 nM T58992 C2B3EM 24822300 Ki = 15.8 nM T58992 C1JRM9 24822458 Ki = 19.91 nM T58992 C5VYZ2 24822459 Ki = 2.07 nM T58992 CIC3L7 24822460 Ki = 24.52 nM T58992 C7O9BN 24822461 Ki = 99 nM T58992 C13MJI 24822630 Ki = 0.79 nM T58992 CJK3I4 24822631 Ki = 5.82 nM T58992 CW2B0R 24822632 Ki = 4.23 nM T58992 CRT19I 24822633 Ki = 6.83 nM T58992 CN6JX5 24822634 Ki = 27.18 nM T58992 CCKO91 24822798 Ki = 56.3 nM T58992 CPN52E 24822799 Ki = 3.8 nM T58992 C58EYR 24822801 Ki = 79.23 nM T58992 CBYW42 24822802 Ki = 12.2 nM T58992 CAK7O3 24822964 Ki = 28 nM T58992 C6R3AE 24822965 Ki = 32.4 nM T58992 CYQ27T 24824634 Ki = 36.94 nM T58992 C6TWH4 24824635 Ki = 1.4 nM T58992 CBPQ24 24824636 Ki = 2.73 nM T58992 CCY7A8 24824637 Ki = 9.72 nM T58992 C9G0CI 24824638 Ki = 12.4 nM T58992 CT0PG3 24828463 Ki = 8830 nM T58992 CTZ0S2 24829369 Ki = 810 nM T58992 CI4W6P 24854099 Ki > 10000 nM T58992 CV6NW8 24854100 Ki = 1140 nM T58992 C5ZCJ9 24854101 Ki > 10000 nM T58992 CZM9I7 24854102 Ki > 10000 nM T58992 CO7LG3 24854177 Ki > 10000 nM T58992 C75WFT 24854178 Ki > 10000 nM T58992 CC5KH6 24854179 Ki > 10000 nM T58992 CL06MB 24854180 Ki = 580 nM T58992 C7ED1M 24854260 Ki = 690 nM T58992 C0I4KH 24854261 Ki > 10000 nM T58992 C2ZUH5 24854262 Ki > 10000 nM T58992 CS3JT4 24854263 Ki > 10000 nM T58992 C53SWQ 24854264 Ki = 1930 nM T58992 C9O5NZ 24857819 IC50 > 1000 nM T58992 CN0T1F 24857820 IC50 > 1000 nM T58992 CIJ83R 24873473 EC50 = 1.2 nM T58992 CK61ND 24886211 Ki > 10000 nM T58992 CDR3T2 24886213 Ki = 5000 nM T58992 CNQ6I4 24894028 IC50 > 10000 nM T58992 CT09XK 24978531 IC50 > 10000 nM T58992 CIY83H 24995848 Ki = 448 nM T58992 CDLW86 25001412 Ki > 1000 nM T58992 CU4C8F 25077980 Ki = 5830 nM T58992 CMR05Y 25079852 IC50 = 4.07 nM T58992 CWZ0X3 25079903 IC50 > 10000 nM T58992 CZ4VA7 25087514 IC50 = 3.97 nM T58992 CW5HS3 25087515 IC50 = 104 nM T58992 C9PVG1 25087516 IC50 = 14.3 nM T58992 C19QSV 25092437 Ki = 149 nM T58992 CUO63Q 25129091 Ki = 150 nM T58992 CEI9L2 25129133 Ki = 0.66 nM T58992 CT9CL8 25129432 Ki = 58 nM T58992 CLW14R 25129434 Ki = 18 nM T58992 CQ36GH 25129435 Ki = 9.3 nM T58992 C2XI7E 25129436 Ki = 11 nM T58992 CT30ZV 25129437 Ki = 330 nM T58992 CM6KY3 25129438 Ki = 480 nM T58992 C5PA3S 25129777 Ki = 1300 nM T58992 C9ELP5 25129778 Ki = 68 nM T58992 C5Q3JF 25129779 Ki = 360 nM T58992 C4DL2M 25129780 Ki = 1.5 nM T58992 C60PHW 25169521 Ki = 5.4 nM T58992 CV3Y7O 25169522 Ki = 580 nM T58992 CICS51 25181445 Ki = 3.162 nM T58992 CG6UT3 25181466 Ki = 1.2 nM T58992 CF6RA5 25190572 Ki = 23175 nM T58992 CPK5D7 25190573 Ki = 15325 nM T58992 CON62K 25190574 Ki = 59420 nM T58992 C6S3WN 25190575 Ki = 5412 nM T58992 CF15AH 25190576 Ki = 8210 nM T58992 CBN1Q0 25190577 Ki = 187050 nM T58992 CKB72D 25190578 Ki = 44025 nM T58992 CZR78G 25190579 Ki = 45335 nM T58992 CF2JK0 25190580 Ki = 192050 nM T58992 CE4R2X 25190581 Ki = 60980 nM T58992 CYC6S0 25190582 Ki = 122080 nM T58992 CE61QB 25190583 Ki = 5612 nM T58992 C9V8MS 25190584 Ki = 28990 nM T58992 C3UV5M 25190585 Ki = 32 nM T58992 CKFI42 25190586 Ki = 868 nM T58992 C5UQX3 25190587 Ki = 955 nM T58992 C5J2WE 25190588 Ki = 1525 nM T58992 CX84WI 25190589 Ki = 759 nM T58992 C5RUI9 25190590 Ki = 933 nM T58992 CQY69C 25190591 Ki = 1136 nM T58992 C8SEQ2 25190592 Ki = 4758 nM T58992 C5BS7N 25190593 Ki = 1033 nM T58992 CE19OU 25190594 Ki = 878 nM T58992 CP5ID6 25190595 Ki = 1535 nM T58992 CO8E4G 25190596 Ki = 2381 nM T58992 CX87HD 25190597 Ki = 3176 nM T58992 CY6CV1 25190598 Ki = 1633 nM T58992 CW5UP9 25190599 Ki = 2270 nM T58992 C1C8VK 25190600 Ki = 1676 nM T58992 CL7Q2F 25190601 Ki = 1080 nM T58992 CD0H5U 25190602 Ki = 445 nM T58992 C8OWC0 25190603 Ki = 370 nM T58992 CH06YU 25190604 Ki = 516 nM T58992 CEJ25L 25190605 Ki = 376 nM T58992 CXD5R8 25190606 Ki = 379 nM T58992 CU6W8O 25190607 Ki = 3103 nM T58992 CWJB54 25190608 Ki = 795 nM T58992 CMHS48 25190609 Ki = 2639 nM T58992 CBL9S4 25190610 Ki = 1298 nM T58992 CZ8Y6L 25190611 Ki = 2064 nM T58992 CL9SN6 25190612 Ki = 5016 nM T58992 C1MGY3 25190613 Ki = 1615 nM T58992 CB1G6M 25190614 Ki = 1951 nM T58992 CJLH27 25190615 Ki = 2340 nM T58992 COE65V 25190616 Ki = 2515 nM T58992 C30VGA 25190617 Ki = 2096 nM T58992 CO7IV2 25190618 Ki = 2879 nM T58992 C8Q7WV 25190619 Ki = 1802 nM T58992 C0G4RJ 25190620 Ki = 2980 nM T58992 C7X4IV 25190621 Ki = 1224 nM T58992 CXG8O3 25190622 Ki = 3948 nM T58992 CD5F6A 25190623 Ki = 2600 nM T58992 CFUD47 25190624 Ki = 1790 nM T58992 C15LIW 25190625 Ki = 1693 nM T58992 C3LEW8 25190626 Ki = 1279 nM T58992 CIDV61 25190627 Ki = 1062 nM T58992 CAGS39 25190628 Ki = 1316 nM T58992 CDS2E6 25190629 Ki = 883 nM T58992 CPW19O 25190630 Ki = 5022 nM T58992 C0SBV7 25207946 Ki = 58 nM T58992 C21OJF 25207948 Ki = 9.5 nM T58992 C0P6CS 25207950 Ki = 140 nM T58992 CN9I8E 25208095 Ki > 500 nM T58992 C5OA1N 25208097 Ki = 168 nM T58992 C59IKP 25208099 Ki = 110 nM T58992 C57UGP 25217787 EC50 = 263 nM T58992 C9BJD3 25232367 Ki = 40.78 nM T58992 CK0F7G 25232539 Ki = 191.98 nM T58992 CGLZ15 25232540 EC50 = 15.2 nM T58992 CHG71D 25232541 Ki = 132.5 nM T58992 CGH3W8 25232542 Ki = 148.2 nM T58992 C8E0RL 25232543 Ki = 3.86 nM T58992 CE6JP0 25232724 Ki = 11.61 nM T58992 C0OU5Y 25232725 Ki = 518.32 nM T58992 C3LHO0 25232727 Ki = 64.46 nM T58992 CO74DE 25233078 Ki = 32.19 nM T58992 CJS1L7 25233081 Ki = 29.26 nM T58992 C1INO6 25233083 Ki = 15.42 nM T58992 C83AVG 25233258 Ki = 186.64 nM T58992 C90OGX 25256781 EC50 = 9 nM T58992 C2XS0Y 25256782 EC50 = 16 nM T58992 CKL48U 25256790 Ki = 117.38 nM T58992 C9NC3W 25257431 Ki = 180 nM T58992 C2GH4L 25257432 Ki = 110 nM T58992 C0EC4L 25257433 Ki = 270 nM T58992 CL2Z7J 42629117 Ki = 1039 nM T58992 C0K9TG 44138064 Ki = 0.025 nM T58992 C15NFW 44138152 Ki = 212 nM T58992 CHW05E 44149909 Ki = 19.1 nM T58992 CFP9S1 44157038 Ki = 5200 nM T58992 CU0PY1 44176456 Ki = 35 nM T58992 C7DR0P 44176458 EC50 = 91 nM T58992 C4ZS5G 44176572 EC50 = 280 nM T58992 CP0WQ3 44177145 Ki = 1 nM T58992 CHJ47Y 44177567 EC50 = 2.5 nM T58992 C1W9PD 44177570 EC50 = 0.1 nM T58992 CHI47S 44177668 Ki = 3.1 nM T58992 C2E1GB 44177669 Ki = 0.46 nM T58992 CD3LH2 44177670 EC50 = 0.2 nM T58992 CX2O9F 44177768 Ki = 13 nM T58992 C8XDQ3 44177770 Ki = 58 nM T58992 CPHW46 44177994 Ki = 0.6 nM T58992 CHAO36 44177995 Ki = 2.9 nM T58992 CVOJ62 44178113 Ki = 0.18 nM T58992 CPQ25W 44181744 Ki = 11510 nM T58992 CX4D3R 44188273 Ki = 5.16 nM T58992 C2XE7Y 44189733 IC50 > 10000 nM T58992 CGA8R1 44189735 IC50 > 10000 nM T58992 C50FOG 44189834 IC50 > 10000 nM T58992 C2AV1K 44190762 IC50 = 1690 nM T58992 CF26JI 44233184 EC50 = 27.54 nM T58992 C67CEB 44233185 Ki = 3.7 nM T58992 CSB84Q 44233410 EC50 = 51.29 nM T58992 CCV87B 44235260 Ki = 765 nM T58992 CV2NB5 44235261 Ki = 1120 nM T58992 C0X3VW 44235262 Ki = 6650 nM T58992 C2HM9V 44235488 EC50 = 65 nM T58992 CCO7H6 44235489 Ki > 10000 nM T58992 CW7NH4 44235490 EC50 = 10 nM T58992 C6NIL8 44235491 Ki = 1790 nM T58992 CG9QD7 44240971 Ki = 6.7 nM T58992 CR61KZ 44240972 Ki = 9.2 nM T58992 C0AL2R 44241022 Ki = 14 nM T58992 CK5T9S 44241023 Ki = 59 nM T58992 C6D0HY 44241024 Ki = 47 nM T58992 C5G6DN 44241123 Ki = 0.18 nM T58992 CC63QX 44247589 Ki = 3347 nM T58992 C1O8LH 44253973 Ki = 56 nM T58992 CQN6W3 44253974 Ki = 1400 nM T58992 C47RZO 44254057 Ki = 0.93 nM T58992 C41MNG 44254058 Ki = 1.5 nM T58992 C2SVL6 44254059 Ki = 20 nM T58992 CVW13I 44254060 Ki = 6.9 nM T58992 C0NZW8 44254061 Ki = 11 nM T58992 C3N2KB 44254062 Ki = 3.3 nM T58992 CJW3P2 44254063 Ki = 2.4 nM T58992 C6OJS0 44254504 Ki = 13 nM T58992 CSBD48 44254505 Ki = 10 nM T58992 C1IPQ6 44254506 Ki = 27 nM T58992 CTL57U 44254584 Ki = 50 nM T58992 CZY2S1 44254585 Ki = 18 nM T58992 C9SQ8D 44254859 Ki = 18 nM T58992 CB47EJ 44254954 Ki = 1.2 nM T58992 C79QBX 44254955 Ki = 15 nM T58992 CVCP62 44254956 Ki = 0.53 nM T58992 CK7B1Q 44254957 Ki = 8.1 nM T58992 CJH6K5 44255041 Ki = 18 nM T58992 C5Z9KH 44255042 Ki = 29 nM T58992 C1FE8D 44255043 Ki = 4.6 nM T58992 CGB3A7 44255044 Ki = 1.2 nM T58992 CTY9U6 44255045 Ki = 13 nM T58992 C8HI7P 44256416 Ki = 91.5 nM T58992 C67DCW 44268589 EC50 = 21 nM T58992 CJ7FW4 44269673 IC50 = 910 nM T58992 C8S0VL 44269677 IC50 = 12 nM T58992 C3LQ1G 44269678 IC50 = 1710 nM T58992 C1LOV8 44269681 IC50 = 150 nM T58992 CT4B3Y 44269682 IC50 = 130 nM T58992 C7ILE4 44269730 IC50 = 3290 nM T58992 C14NWL 44269731 IC50 = 870 nM T58992 CMS9P2 44269732 IC50 = 1800 nM T58992 CPF7M8 44269737 IC50 = 1970 nM T58992 C82YGV 44269750 IC50 = 1.15 nM T58992 C1SJ0O 44269751 IC50 = 560 nM T58992 CB7D3I 44269752 IC50 = 50 nM T58992 C4PG9V 44269757 IC50 > 10000 nM T58992 CW75BD 44269767 IC50 > 10000 nM T58992 CY61IX 44269822 IC50 > 10000 nM T58992 CW7C4R 44269855 IC50 > 10000 nM T58992 CUH74K 44269856 IC50 > 10000 nM T58992 CMIZ34 44269859 IC50 > 10000 nM T58992 CG93NF 44269868 IC50 > 10000 nM T58992 CE26RM 44269871 IC50 > 10000 nM T58992 C35VDR 44269872 IC50 > 10000 nM T58992 C6Y8IM 44269891 IC50 > 10000 nM T58992 C3X2ID 44269895 IC50 > 10000 nM T58992 CM62ZD 44269901 IC50 > 10000 nM T58992 C6T9WO 44269902 IC50 > 10000 nM T58992 CQ2W3Z 44269927 IC50 > 10000 nM T58992 C2CAI8 44269932 IC50 = 5600 nM T58992 CJQI23 44269933 IC50 > 10000 nM T58992 C8AMT3 44269936 IC50 > 10000 nM T58992 C9H0AG 44269950 IC50 > 10000 nM T58992 CQ20KW 44269951 IC50 > 10000 nM T58992 C89YQU 44269952 IC50 > 10000 nM T58992 C0H4SW 44269967 IC50 > 10000 nM T58992 CZ49TF 44269969 IC50 > 10000 nM T58992 CTRE60 44269980 IC50 > 10000 nM T58992 CIFJ07 44269988 IC50 > 10000 nM T58992 CWU8M4 44269994 IC50 = 460 nM T58992 CAG2N4 44270012 IC50 > 10000 nM T58992 CP4C3N 44272933 Ki = 4100 nM T58992 C0XJC1 44272934 Ki = 1600 nM T58992 CBRV50 44273019 Ki = 28 nM T58992 COAK72 44273020 Ki = 180 nM T58992 CO3CK8 44273021 Ki = 48 nM T58992 CXPK83 44273048 Ki = 1300 nM T58992 CHR3A4 44273049 Ki = 1900 nM T58992 C6DGE7 44273050 Ki = 3300 nM T58992 CB35OI 44273081 Ki = 22 nM T58992 CW2E6Z 44273082 Ki = 8.2 nM T58992 C7Z5NO 44273237 Ki > 100000 nM T58992 CRN21P 44273377 Ki = 150 nM T58992 C2CEN5 44273397 Ki = 1.1 nM T58992 CR2S9J 44273399 Ki = 1 nM T58992 C1TS8N 44273477 Ki = 3.7 nM T58992 CW5RT0 44273569 Ki = 6.5 nM T58992 C7ON5L 44273683 Ki = 3.1 nM T58992 C5V8TG 44274454 Ki = 703 nM T58992 CW36SV 44274467 Ki = 1073 nM T58992 CI0K5N 44274481 Ki = 135 nM T58992 CFLU92 44274482 Ki = 4.79 nM T58992 C7NQW1 44274561 Ki = 49.7 nM T58992 CS15FN 44274614 Ki = 62.4 nM T58992 CUY91K 44274615 Ki = 1.38 nM T58992 C6M3CV 44275470 IC50 = 1904 nM T58992 CSJ5D4 44275471 IC50 = 1394 nM T58992 C5X0ID 44275484 IC50 = 44.3 nM T58992 C42JFC 44275507 IC50 = 1724 nM T58992 CI4S9N 44275523 IC50 = 2600 nM T58992 CDLO89 44275536 IC50 = 500 nM T58992 C2HZ7J 44275550 IC50 = 7.2 nM T58992 CUR4J2 44275566 IC50 = 607 nM T58992 CUL53A 44275567 IC50 = 360 nM T58992 C0DSJ6 44275568 IC50 = 82.4 nM T58992 CK3MP0 44275684 IC50 = 4 nM T58992 CW0G2J 44275878 IC50 = 250 nM T58992 CU9E1H 44275879 IC50 = 8097 nM T58992 C7BZ1U 44275996 IC50 = 13 nM T58992 C2M3DV 44276013 IC50 = 1.4 nM T58992 C4B9HA 44276027 IC50 = 120 nM T58992 C7SE0I 44276028 IC50 = 5.8 nM T58992 CSN06P 44276042 IC50 = 5.5 nM T58992 C54XUF 44276048 IC50 = 11.4 nM T58992 CC6L1Z 44276066 IC50 = 10 nM T58992 CB7V1Y 44276158 IC50 = 42 nM T58992 CFAB48 44276159 IC50 = 29 nM T58992 C9LXY8 44276213 Ki = 4.2 nM T58992 CU7E8G 44276236 IC50 = 845 nM T58992 C43NLT 44276269 Ki = 0.019 nM T58992 C43UHA 44276278 IC50 = 1.8 nM T58992 C8OS7J 44276292 Ki = 2 nM T58992 C58VFX 44276293 Ki = 5 nM T58992 CW6P4Y 44276782 Ki > 10000 nM T58992 CC2OD4 44278111 Ki > 10000 nM T58992 CRMA84 44278114 Ki > 10000 nM T58992 CF0Y4M 44278115 Ki > 10000 nM T58992 CUS04C 44279592 Ki = 5.52 nM T58992 CL70JN 44279594 Ki = 8.47 nM T58992 C3AYK9 44279686 EC50 = 1.1 nM T58992 C9STZ5 44279699 EC50 = 0.3 nM T58992 C5A4FH 44282798 Ki = 11 nM T58992 CK3JH6 44283842 Ki = 37 nM T58992 CUGL03 44283843 Ki = 117 nM T58992 CX9KP8 44284742 Ki = 420 nM T58992 CWKT78 44285029 Ki > 500 nM T58992 CQ15BW 44285070 Ki > 500 nM T58992 CSI6F5 44285718 Ki = 0.74 nM T58992 CN7V6X 44286598 Ki = 205 nM T58992 CV46BG 44286647 Ki = 127 nM T58992 C69JKC 44286719 Ki = 263 nM T58992 CY9PS5 44286720 Ki = 113 nM T58992 C6QZ4H 44286867 IC50 = 0.53 nM T58992 C6NQ5U 44286870 Ki > 1000 nM T58992 C6SJY9 44286875 IC50 = 177 nM T58992 C4CYJ1 44286876 IC50 = 45 nM T58992 C41IRN 44286883 Ki = 159 nM T58992 CNOB73 44286884 Ki = 649 nM T58992 C7SZ0Y 44286885 Ki = 52.7 nM T58992 C3JRH1 44286895 IC50 = 178 nM T58992 CS54YC 44287020 IC50 = 10.7 nM T58992 CHU57Z 44287142 Ki = 554 nM T58992 C39XJE 44287143 Ki = 330 nM T58992 C2Y3MA 44287144 IC50 = 1.6 nM T58992 CRO32K 44287168 Ki > 1000 nM T58992 C09XZL 44287189 Ki = 509 nM T58992 CW9TN6 44287225 IC50 = 24 nM T58992 C8U5QT 44287236 Ki = 308 nM T58992 C0RE2U 44287369 Ki = 551 nM T58992 CL6K5U 44287383 Ki > 1000 nM T58992 CQ46MS 44287394 Ki = 443 nM T58992 CQU8Z1 44287414 Ki = 508 nM T58992 C7M2FV 44287415 Ki > 1000 nM T58992 C1RE2J 44287486 Ki = 113 nM T58992 C97UNH 44287487 Ki = 140 nM T58992 C9DZE3 44291256 Ki = 49 nM T58992 CV9F0L 44291264 Ki = 290 nM T58992 CQI1R7 44291332 Ki = 330 nM T58992 C1M2TF 44291354 Ki > 750 nM T58992 C7IY6S 44291655 Ki = 46 nM T58992 C5WE4Y 44292142 IC50 = 1160 nM T58992 CE3YS4 44292200 IC50 = 52 nM T58992 C0VR9X 44292280 IC50 = 10.9 nM T58992 CIEU38 44292281 IC50 = 236 nM T58992 CARS41 44292403 IC50 = 1520 nM T58992 C2ST7W 44292414 IC50 = 13.5 nM T58992 C3KYZ5 44292426 IC50 = 52.7 nM T58992 C2ET5R 44292437 IC50 = 2540 nM T58992 C31UAT 44292682 Ki > 10000 nM T58992 CS9QC6 44292684 Ki > 10000 nM T58992 CR48ED 44292854 Ki = 14 nM T58992 C04APC 44292946 Ki = 9.6 nM T58992 CF5TP9 44292986 Ki = 1900 nM T58992 CK5R2O 44292987 Ki = 5 nM T58992 CSC5V1 44293140 Ki > 1000 nM T58992 C6MQ8U 44295810 Ki > 100 nM T58992 CUAR49 44296549 Ki = 853 nM T58992 CD3EK7 44296582 Ki = 2409 nM T58992 CACV07 44297100 Ki = 183 nM T58992 C1V4OE 44297195 Ki = 1.24 nM T58992 C9AF6B 44297435 Ki = 2075 nM T58992 CNP5W1 44297519 Ki > 10000 nM T58992 C9UY4E 44297697 Ki = 1838 nM T58992 C8F1ST 44297727 Ki > 10000 nM T58992 C3QR5B 44298187 Ki = 12 nM T58992 COR8C1 44298198 Ki = 19 nM T58992 CSA32D 44298201 Ki = 570 nM T58992 C91RLI 44298202 Ki = 250 nM T58992 CN7CO4 44298203 Ki = 2800 nM T58992 CMN0R9 44298206 Ki = 1800 nM T58992 CX2EQ7 44298207 Ki = 810 nM T58992 CS49XN 44298213 Ki = 3600 nM T58992 C9QLX2 44298221 Ki = 160 nM T58992 C9BQY0 44298233 Ki = 470 nM T58992 CO8K1I 44298240 Ki = 460 nM T58992 C4YG5R 44298841 Ki > 10000 nM T58992 CF8YG9 44299258 Ki = 32 nM T58992 C7ZYM4 44299404 EC50 = 0.14 nM T58992 C5BW6K 44299840 Ki = 1700 nM T58992 CTB24D 44299841 Ki = 1400 nM T58992 CIXY54 44299842 Ki = 880 nM T58992 CT6HW3 44300146 Ki = 9.8 nM T58992 CIQ4Z8 44300188 Ki = 420 nM T58992 C1Q7TB 44300209 Ki = 52 nM T58992 CQWA30 44300211 Ki = 2400 nM T58992 C6X2TZ 44300212 Ki = 6200 nM T58992 C90DFQ 44300216 Ki = 37 nM T58992 C4GY1Z 44300227 Ki > 10000 nM T58992 CV08SA 44300800 Ki = 578 nM T58992 C9IL2D 44301524 Ki = 154.88 nM T58992 CY69XZ 44301533 Ki > 10000 nM T58992 C4CKF2 44301534 Ki = 10000 nM T58992 CT1R7F 44301641 Ki = 1400 nM T58992 C0LZ1I 44301653 Ki > 1000000 nM T58992 C9PEI7 44301663 Ki = 170 nM T58992 CJ1W3X 44301664 Ki > 10000 nM T58992 CG6JI1 44301701 EC50 = 1.7 nM T58992 CGK5F3 44301963 Ki > 1000000 nM T58992 C4ASQ5 44302312 Ki = 459 nM T58992 C91ALC 44302324 Ki = 863 nM T58992 C9MP0A 44302743 Ki = 87.8 nM T58992 C26CLF 44302821 IC50 > 10000 nM T58992 CD47TR 44302918 Ki = 47.2 nM T58992 CNI7U6 44302972 IC50 > 10000 nM T58992 CL6I9X 44302973 IC50 > 10000 nM T58992 CB2H7L 44302988 IC50 > 10000 nM T58992 C28OYR 44302993 IC50 > 10000 nM T58992 C23GUZ 44303030 IC50 > 10000 nM T58992 CWM93O 44303041 IC50 = 5214 nM T58992 C4VN8H 44303094 IC50 > 10000 nM T58992 C2RTS0 44303112 IC50 > 10000 nM T58992 CGS81I 44303376 IC50 > 10000 nM T58992 CXN7F0 44303379 IC50 > 10000 nM T58992 CICN21 44303386 IC50 = 4350 nM T58992 C2L9UZ 44303682 IC50 > 10000 nM T58992 C1CI7Y 44303692 IC50 = 639 nM T58992 CAH1C5 44306509 IC50 = 740 nM T58992 CAL02W 44306565 Ki = 13.16 nM T58992 CT7SC8 44306566 Ki = 1.45 nM T58992 CHKQ16 44306567 Ki = 2.24 nM T58992 CR56FX 44306606 Ki = 5.48 nM T58992 CUHK45 44306640 Ki = 2.09 nM T58992 CY0HT8 44306645 Ki = 38.97 nM T58992 C0TKD8 44306682 Ki = 6.39 nM T58992 C5G7IS 44306729 Ki = 49.3 nM T58992 CX8UW1 44306748 Ki = 4.14 nM T58992 CTMU85 44306771 Ki = 6.66 nM T58992 C1VG3T 44306787 Ki = 0.51 nM T58992 CWT5Q7 44306866 Ki = 24 nM T58992 CXG6D2 44306867 Ki = 407 nM T58992 CSA9Y2 44306943 Ki = 1.59 nM T58992 CMR0I7 44306944 Ki = 22 nM T58992 C1IBV3 44306952 Ki = 27.24 nM T58992 CEK0S4 44306977 Ki = 0.72 nM T58992 CB9P4T 44306987 Ki = 5.9 nM T58992 C4ZU1Q 44306988 Ki = 1.89 nM T58992 CUE6H5 44307017 Ki = 20.77 nM T58992 CZX25T 44307027 Ki = 4.5 nM T58992 CMU50G 44307036 Ki = 63.4 nM T58992 C9SEL1 44307066 Ki = 0.86 nM T58992 CB74GN 44307067 Ki = 3.88 nM T58992 C3WRJ5 44307068 Ki = 26.17 nM T58992 C7K4VR 44307116 Ki = 12.3 nM T58992 CW5BN2 44307131 Ki = 16.61 nM T58992 CTV0Q4 44307157 Ki = 11.29 nM T58992 CH0YD7 44307168 Ki = 29.63 nM T58992 CRTW95 44307176 Ki = 0.384 nM T58992 CRMH14 44307182 Ki = 5.67 nM T58992 C0X3HL 44307191 Ki = 8.3 nM T58992 CW9JX4 44307198 Ki = 19.79 nM T58992 CM6J0K 44307210 Ki = 7.8 nM T58992 CY1H2U 44307211 Ki = 1.32 nM T58992 CQ2HL0 44307228 Ki = 0.93 nM T58992 C4E3GT 44307234 Ki = 23.62 nM T58992 COS3X0 44307318 Ki = 53.86 nM T58992 C82AYR 44307326 Ki = 2.02 nM T58992 CTX9O8 44307330 Ki = 13 nM T58992 CI8XV3 44307356 Ki = 1.36 nM T58992 CC7F4Q 44307381 Ki = 15.9 nM T58992 C5G2VA 44307382 Ki = 23.7 nM T58992 CCN57J 44307428 Ki = 0.25 nM T58992 C0GJT5 44311043 Ki = 53 nM T58992 C2GE8X 44311351 Ki = 75 nM T58992 CV9X4Q 44311893 Ki = 3.31 nM T58992 C9KO7E 44311978 Ki = 5.5 nM T58992 CLX5V8 44312109 Ki = 3.79 nM T58992 C75XAK 44312914 Ki = 85.7 nM T58992 CX2S3L 44316421 IC50 = 49100 nM T58992 C10ESM 44316464 IC50 = 3400 nM T58992 CH1M5U 44316465 IC50 > 100000 nM T58992 C9W8IB 44316466 IC50 = 7180 nM T58992 COH84N 44316561 IC50 = 6610 nM T58992 CW1I9R 44316562 IC50 = 600000 nM T58992 C6CN0Q 44316570 IC50 = 90000 nM T58992 C9Z5RH 44316576 IC50 > 100000 nM T58992 CF7E3Y 44316678 IC50 = 24600 nM T58992 CZYD37 44316856 IC50 = 431 nM T58992 CDE7W8 44318784 IC50 = 7400 nM T58992 C3KE8A 44319002 IC50 = 7900 nM T58992 C4HUA9 44323614 Ki = 9.35 nM T58992 CM0G8A 44324324 Ki = 6800 nM T58992 CALT96 44324339 Ki = 3900 nM T58992 C2Y4SJ 44324361 Ki = 8800 nM T58992 CT39YA 44324362 Ki = 7100 nM T58992 CDX6T3 44325124 Ki = 69 nM T58992 CZGQ80 44325125 Ki = 5.6 nM T58992 CR0G2S 44325129 Ki = 5.6 nM T58992 CAKF25 44325133 Ki = 0.54 nM T58992 CCWZ94 44325134 Ki = 4.1 nM T58992 C3E0LY 44325135 Ki = 10 nM T58992 CC2I6S 44325138 Ki = 0.85 nM T58992 COEW46 44325139 Ki = 6.9 nM T58992 CBJQ30 44325180 Ki = 27 nM T58992 CC42YP 44325181 Ki = 42 nM T58992 C7I5JO 44325202 Ki = 110 nM T58992 CTA3S5 44325215 Ki = 29 nM T58992 C4M7AE 44325216 Ki = 33 nM T58992 CVI70N 44325318 Ki = 130 nM T58992 CBAF64 44325319 Ki = 51 nM T58992 CU6A7N 44325320 Ki = 8.5 nM T58992 C4PY5Q 44325444 Ki = 420 nM T58992 C05WRM 44325455 Ki = 3.1 nM T58992 C0GR8Q 44325457 Ki = 23 nM T58992 C76RSH 44325483 Ki = 3.1 nM T58992 CIQ2U7 44325484 Ki = 2.6 nM T58992 CY9BC0 44326368 IC50 = 16 nM T58992 C0BR8P 44326371 IC50 = 21 nM T58992 C0FUD3 44326372 IC50 = 29 nM T58992 C7F8TX 44326413 IC50 = 30 nM T58992 CE9W0C 44326414 IC50 = 71 nM T58992 CE69ON 44326415 IC50 = 15 nM T58992 CY1ML0 44326426 IC50 = 46 nM T58992 CR8K3D 44326480 Ki = 21.38 nM T58992 CC87GE 44328387 Ki = 2.1 nM T58992 CTU26X 44328406 Ki = 9.3 nM T58992 CV61EB 44328435 Ki = 0.96 nM T58992 C5NHT1 44329096 Ki = 16 nM T58992 CV57DK 44329162 Ki = 40 nM T58992 C8ABT2 44329206 Ki = 500 nM T58992 CH46CQ 44329417 Ki = 210 nM T58992 CV91DR 44329508 Ki = 44 nM T58992 CL3B0J 44329509 Ki = 41 nM T58992 C1LOP6 44329524 Ki = 260 nM T58992 C2JOC8 44329698 Ki = 8.2 nM T58992 CV90JY 44329722 Ki = 4.7 nM T58992 C9YU3Z 44329726 Ki > 7200 nM T58992 COE92S 44329727 Ki = 3400 nM T58992 COR3H8 44329728 Ki = 2400 nM T58992 C0UBK2 44331831 IC50 = 2.44 nM T58992 C8RC7M 44331854 IC50 = 0.69 nM T58992 CL4H2F 44331862 IC50 = 0.32 nM T58992 CREU72 44331873 IC50 = 0.71 nM T58992 CR0UZ9 44333058 Ki = 12.2 nM T58992 C2U3XV 44334636 Ki = 21.4 nM T58992 CF81BW 44334658 Ki = 25.6 nM T58992 CPA67X 44334707 Ki = 42 nM T58992 C89MXB 44335064 Ki = 334 nM T58992 CJG5O0 44335120 Ki = 13.8 nM T58992 C26IAM 44336365 Ki = 2 nM T58992 CWQ04R 44336430 Ki = 9.5 nM T58992 C24UOF 44336449 Ki = 84 nM T58992 CJ4WL1 44336602 Ki = 420 nM T58992 CGZ9N2 44336905 Ki = 2923 nM T58992 CDJ9C5 44336988 IC50 = 45.5 nM T58992 CYMH75 44337108 Ki = 2709 nM T58992 CJ0I6Q 44337123 Ki = 4787 nM T58992 CPOX86 44337129 Ki = 7722 nM T58992 CT78UG 44337131 Ki = 3312 nM T58992 CKGS32 44337160 IC50 = 672 nM T58992 CO8Y5G 44337163 Ki = 8819 nM T58992 CWJC16 44337164 IC50 = 24.7 nM T58992 CBJ01F 44337212 Ki = 11240 nM T58992 C8IJM5 44337229 Ki = 8710 nM T58992 C97YKG 44337230 Ki = 39120 nM T58992 C3B4WO 44337231 Ki = 5011 nM T58992 CU8IY3 44337232 Ki = 4987 nM T58992 C3GQ1S 44337243 IC50 = 542 nM T58992 C3M0QX 44337249 Ki = 12270 nM T58992 C0MJL2 44337252 Ki = 31780 nM T58992 CVE93R 44337264 IC50 > 1000 nM T58992 CL27XI 44337269 IC50 = 19.7 nM T58992 CVS69U 44337271 IC50 = 50.9 nM T58992 C14LMK 44337273 IC50 = 25.9 nM T58992 CM5YJ1 44337274 IC50 = 22.6 nM T58992 C0XI3O 44337275 IC50 = 10.7 nM T58992 C5D6QW 44337276 IC50 = 106 nM T58992 CB1U3P 44337314 IC50 = 54 nM T58992 CPHU86 44337316 IC50 = 374 nM T58992 CU35AM 44337344 IC50 = 4.35 nM T58992 CB85KA 44337351 Ki = 22370 nM T58992 CI13YG 44337357 Ki = 1439 nM T58992 CW2FZ7 44337362 Ki = 2919 nM T58992 CJ08FM 44337379 Ki = 8048 nM T58992 CO90UJ 44337393 Ki > 10000 nM T58992 C2EB8Z 44337394 Ki = 141 nM T58992 CRD71H 44337420 Ki > 10000 nM T58992 CIP87K 44337437 Ki = 3913 nM T58992 CG65HU 44337443 Ki = 95 nM T58992 CEDX21 44337444 Ki = 209 nM T58992 CR62KO 44337452 Ki = 16460 nM T58992 C9CIP3 44337459 Ki = 5013 nM T58992 CFA2Q7 44337460 Ki = 7430 nM T58992 CF96JK 44337473 Ki = 10090 nM T58992 CX87AS 44337513 Ki = 7579 nM T58992 CP1VN3 44337550 Ki = 4978 nM T58992 CZ02BO 44337551 Ki = 5958 nM T58992 CIZA68 44337576 Ki = 229 nM T58992 C59YHG 44337591 Ki = 67 nM T58992 C4AIE7 44337613 EC50 = 4.19 nM T58992 CHB64V 44337616 Ki = 2.25 nM T58992 C35PQC 44337617 Ki = 2.6 nM T58992 CKZ03N 44337618 Ki = 2.43 nM T58992 C7A9FQ 44337642 Ki = 51.4 nM T58992 C6AVW4 44337643 Ki = 7.41 nM T58992 C8OFG5 44337644 Ki = 59.45 nM T58992 C59RIN 44337645 Ki = 103 nM T58992 C18MWY 44337673 Ki = 3.12 nM T58992 CI8AT5 44337683 Ki = 5.66 nM T58992 C0J9UR 44337749 Ki = 11.19 nM T58992 CJTU61 44337750 Ki = 70.15 nM T58992 CMGC86 44337764 Ki = 21.76 nM T58992 CI48SV 44337765 Ki = 7.67 nM T58992 CVP73N 44337783 Ki = 5.29 nM T58992 C7Q4HS 44337789 Ki = 15.9 nM T58992 CP4A0K 44337800 Ki = 23.2 nM T58992 C64JKH 44337822 Ki = 7.33 nM T58992 C20HGO 44337823 Ki = 17.02 nM T58992 C40VWE 44337830 Ki = 27.56 nM T58992 C3QGP4 44337831 Ki = 20.1 nM T58992 CHVG85 44337832 Ki = 3.53 nM T58992 CS57JZ 44337839 Ki = 82.5 nM T58992 C9CIL3 44339409 EC50 = 86.8 nM T58992 CFNR91 44339423 Ki = 10000 nM T58992 CW56BK 44339424 Ki = 5674 nM T58992 CF1HE6 44339472 EC50 = 1613 nM T58992 CFRJ92 44339475 EC50 = 7.91 nM T58992 C68ZSO 44339521 EC50 = 20.6 nM T58992 CX93QM 44339562 Ki = 11.7 nM T58992 CO9IF8 44339563 Ki = 0.322 nM T58992 C7E4MS 44339576 Ki = 8779 nM T58992 C34DEN 44339684 Ki = 10000 nM T58992 CO3C7M 44339695 Ki = 10000 nM T58992 CM42BN 44341722 Ki = 19.06 nM T58992 CND5T9 44341920 Ki = 18.99 nM T58992 CM4NE8 44342057 IC50 = 620 nM T58992 C6BX2A 44342141 IC50 > 10000 nM T58992 CD9ZS8 44342270 IC50 = 1410 nM T58992 C4N6GE 44342597 Ki = 464 nM T58992 C0Z9DY 44342598 Ki = 114 nM T58992 CSZ34A 44342661 Ki = 57 nM T58992 CJVN97 44342684 Ki = 2934 nM T58992 CP97HW 44342724 Ki = 7000 nM T58992 C2EQZ1 44342741 Ki = 7000 nM T58992 CYTQ61 44342743 Ki = 788 nM T58992 C0IJN7 44342746 Ki = 1586 nM T58992 CQ5B8R 44342747 Ki = 2584 nM T58992 CW5RB3 44342753 Ki = 7000 nM T58992 C1LQR9 44342754 Ki = 7000 nM T58992 CD3F2N 44342792 Ki = 7000 nM T58992 CC1X5F 44342793 Ki = 7000 nM T58992 C46PTB 44342843 Ki = 4200 nM T58992 CNO76C 44342910 Ki = 152 nM T58992 C5NQP9 44342911 Ki = 37 nM T58992 CNG79I 44342912 Ki = 98 nM T58992 CLC0Z1 44342925 Ki = 67 nM T58992 C74GDW 44342933 Ki = 78 nM T58992 CG1X6K 44342934 Ki = 158 nM T58992 C0YV2K 44346065 Ki = 53.2 nM T58992 CNPW90 44348435 IC50 > 10 nM T58992 CI05WF 44348542 IC50 > 10 nM T58992 C0JWA6 44348797 IC50 = 2066 nM T58992 CPV8R3 44349947 Ki = 15.3 nM T58992 C9C3IY 44350380 IC50 = 1653 nM T58992 CN4TR3 44350651 IC50 = 390 nM T58992 CR47MU 44350667 IC50 = 1370 nM T58992 CB81CH 44350794 IC50 = 1908 nM T58992 C5YEQ9 44353390 Ki = 0.3 nM T58992 C0TJQ7 44353391 Ki = 0.015 nM T58992 CFR4W6 44353454 Ki = 0.14 nM T58992 CH93BM 44353457 Ki = 0.00066 nM T58992 CR90GZ 44353458 Ki = 0.083 nM T58992 CW79ZB 44353468 Ki = 0.013 nM T58992 C4OZW5 44354228 Ki = 750 nM T58992 C4HYP6 44355590 Ki = 250 nM T58992 CVO2G3 44355745 Ki = 0.5 nM T58992 CMS4H1 44355747 Ki = 1.6 nM T58992 C8VW0Y 44355787 Ki = 6.8 nM T58992 CK3R5G 44356181 IC50 = 30 nM T58992 C1DQ2G 44357097 Ki = 935 nM T58992 C9QT7R 44358763 Ki = 1200 nM T58992 C1UXN9 44358875 Ki = 310 nM T58992 C84JQO 44358880 Ki = 14 nM T58992 CD2KB4 44358890 Ki = 73 nM T58992 CG7H8O 44358892 Ki = 110 nM T58992 C5R1NH 44358904 Ki = 57 nM T58992 C1JUA9 44358924 Ki = 220 nM T58992 CG68ZO 44358969 Ki = 270 nM T58992 C1F3PX 44361303 Ki = 176 nM T58992 CW2RE7 44361306 Ki = 449 nM T58992 C6QKO2 44361311 Ki = 558 nM T58992 C2YLK0 44365777 Ki = 1.48 nM T58992 C3ZS6Q 44366280 Ki > 10000 nM T58992 C1C3WO 44366432 Ki > 10000 nM T58992 CU8MZ9 44366433 Ki > 10000 nM T58992 CD18TR 44366689 Ki = 10900 nM T58992 CYL95J 44366690 Ki = 7050 nM T58992 C7IFR8 44366822 Ki = 222 nM T58992 CL1JV2 44366823 Ki = 5200 nM T58992 COEC43 44367007 Ki = 322 nM T58992 CTY04M 44367017 Ki = 2.7 nM T58992 CT71JB 44367028 Ki = 23.5 nM T58992 C30QSI 44367136 Ki = 13.7 nM T58992 C8IZ2L 44367182 EC50 = 41 nM T58992 CRO21Y 44367308 Ki = 21.2 nM T58992 C8BX2S 44367339 Ki = 17.3 nM T58992 CF5Q6M 44368739 Ki = 12.2 nM T58992 CJA53V 44369365 IC50 = 35 nM T58992 C63ZIN 44369383 IC50 = 12 nM T58992 C8BU7I 44369600 IC50 = 21 nM T58992 C5QFT8 44369609 IC50 = 22 nM T58992 CA8I2T 44369628 IC50 = 1.8 nM T58992 CJN80S 44369629 IC50 = 6.5 nM T58992 CYA9W4 44369919 IC50 = 25.5 nM T58992 C2SL0X 44371817 Ki = 320 nM T58992 C9YU5O 44371818 Ki = 59 nM T58992 CJRF15 44371877 Ki > 35000 nM T58992 CIGL43 44371878 Ki = 63 nM T58992 CWJ7E2 44371894 Ki = 2700 nM T58992 C79VFD 44371907 Ki = 570 nM T58992 C9XK2F 44374175 Ki = 230 nM T58992 CF9Z8Q 44374177 Ki = 123 nM T58992 C13FDT 44374197 Ki = 46 nM T58992 CRZ03M 44374199 Ki = 36 nM T58992 CXM2W1 44374294 Ki = 85 nM T58992 C95JYL 44374319 Ki = 25000 nM T58992 CBPG98 44374358 Ki = 66 nM T58992 C6AJ1E 44374448 Ki = 119 nM T58992 CNI91A 44374450 Ki = 26 nM T58992 CMAZ21 44377350 IC50 = 1.93 nM T58992 CAEZ31 44377417 Ki = 2.4 nM T58992 C30LNT 44377418 Ki = 17 nM T58992 CGWR19 44377496 Ki = 4.6 nM T58992 CZ1C5I 44377510 IC50 = 31.2 nM T58992 CEN28I 44377511 IC50 = 389 nM T58992 C3K1LP 44377512 IC50 = 107 nM T58992 C5FD0K 44377582 IC50 = 82.5 nM T58992 CS39DL 44377583 IC50 = 86.3 nM T58992 C3NIQ7 44377592 Ki = 47 nM T58992 C20KEA 44377655 Ki = 75 nM T58992 CM67GP 44377678 Ki = 39 nM T58992 CW3MA7 44377703 IC50 = 9.6 nM T58992 C89OJS 44377704 IC50 = 6.54 nM T58992 CZAQ72 44377733 Ki = 16 nM T58992 C6PK2H 44377757 Ki = 0.7 nM T58992 C9FZI2 44380063 Ki = 1.3 nM T58992 CWAU81 44380064 Ki = 0.7 nM T58992 CAY94G 44380352 Ki = 0.8 nM T58992 CP0GX5 44380353 Ki = 0.6 nM T58992 C0FVP6 44380370 Ki = 1.2 nM T58992 C7XG9B 44380504 Ki = 1.1 nM T58992 CW6UE7 44380600 Ki = 4.4 nM T58992 CRWH28 44380931 Ki = 220 nM T58992 CE0C5H 44380980 Ki = 20 nM T58992 CT84GR 44380994 Ki = 37 nM T58992 CO8W9Y 44381023 Ki = 11 nM T58992 C4AX6I 44381041 Ki = 80 nM T58992 CM6Y4U 44381048 Ki = 240 nM T58992 CB26OS 44381112 Ki = 21 nM T58992 CLA45Q 44381243 Ki = 170 nM T58992 CK8SV3 44381244 Ki = 250 nM T58992 CJ4K2P 44381335 Ki = 8.3 nM T58992 C98GKV 44381336 Ki = 6.2 nM T58992 C6P9IF 44381337 Ki = 26 nM T58992 CFHB60 44381349 Ki = 29 nM T58992 CO80DQ 44381356 Ki = 75 nM T58992 CA34PO 44381357 Ki = 180 nM T58992 CP86KQ 44381360 Ki = 100 nM T58992 CX94ZT 44381517 Ki = 61 nM T58992 CB3T2V 44381518 Ki = 98 nM T58992 CM72XA 44381519 Ki = 13 nM T58992 CU4X6R 44383702 Ki = 10.1 nM T58992 CM2C7Z 44383840 Ki = 12.9 nM T58992 C53YNW 44383845 Ki = 2.66 nM T58992 C86HYE 44383903 Ki = 0.77 nM T58992 CQM6T1 44383911 Ki = 0.82 nM T58992 CUAV19 44383955 Ki = 2.41 nM T58992 CA18YP 44383956 Ki = 27.4 nM T58992 CK1P0O 44384018 Ki = 0.55 nM T58992 C6CJ0X 44384062 Ki = 19 nM T58992 CS60NH 44384534 Ki = 1.78 nM T58992 CBKJ02 44385119 Ki = 381 nM T58992 CS2J1L 44385163 Ki = 0.89 nM T58992 CA9ET7 44385170 Ki = 0.24 nM T58992 CBCX28 44385172 Ki = 6.44 nM T58992 CEG10S 44385238 Ki = 0.4 nM T58992 CL2KH8 44385239 Ki = 0.44 nM T58992 C4PZX7 44385245 Ki = 0.26 nM T58992 CD4L2B 44385830 Ki = 281 nM T58992 CXQ19H 44386782 IC50 = 11.62 nM T58992 C5ZFX2 44394283 Ki > 2000 nM T58992 COB70L 44394284 Ki > 2000 nM T58992 C5BTZ1 44394320 Ki > 2000 nM T58992 C6DB4X 44394324 Ki > 2000 nM T58992 C2OV9B 44394344 Ki > 2000 nM T58992 C1Y3NV 44394345 Ki > 2000 nM T58992 CCR2U1 44394375 Ki > 2000 nM T58992 CQ2O6J 44394381 Ki > 2000 nM T58992 CTJ2I9 44394405 Ki > 2000 nM T58992 CLFU54 44394419 Ki > 2000 nM T58992 C0A1OW 44394487 Ki > 2000 nM T58992 C61AXY 44394529 Ki > 2000 nM T58992 CRCV49 44394559 Ki > 2000 nM T58992 CV8JF2 44396503 EC50 = 82 nM T58992 CL6WV3 44398138 Ki > 10000 nM T58992 CJ98TY 44398175 Ki = 4820 nM T58992 C56JOK 44399274 Ki = 900 nM T58992 CC1UY9 44399493 Ki = 173 nM T58992 C4XEQ2 44399584 Ki = 898 nM T58992 CR0G7H 44399648 Ki = 55 nM T58992 CT2YO6 44399674 Ki = 1500 nM T58992 CMA91N 44399675 Ki = 1496 nM T58992 C9GF1J 44399730 Ki = 1300 nM T58992 CXR91I 44401402 Ki = 480 nM T58992 CQRZ78 44401457 Ki = 4.2 nM T58992 C3Y4MD 44401653 Ki = 130 nM T58992 C1B4QL 44403095 Ki > 10000 nM T58992 C1YL7Z 44403098 Ki > 10000 nM T58992 CFV98A 44403101 Ki > 10000 nM T58992 C6OY9S 44403102 Ki > 10000 nM T58992 CH4SX6 44403105 Ki > 10000 nM T58992 C12FIH 44403106 Ki > 10000 nM T58992 C4LKC1 44404394 Ki > 10000 nM T58992 C3EJ4G 44404396 Ki > 10000 nM T58992 CILB28 44404652 IC50 > 10000 nM T58992 CA58SU 44404670 IC50 > 10000 nM T58992 C83PCH 44404679 IC50 > 10000 nM T58992 CU0YX9 44404684 IC50 > 10000 nM T58992 CEJ7F8 44404689 IC50 = 300 nM T58992 CODG94 44404695 IC50 = 8800 nM T58992 CD79WM 44404698 IC50 = 9400 nM T58992 C0BED6 44404699 IC50 > 10000 nM T58992 C2NHS0 44404707 IC50 = 5700 nM T58992 CNX5T8 44404731 IC50 > 10000 nM T58992 CN0G4K 44405139 Ki > 5000 nM T58992 CE81GQ 44405140 Ki > 5000 nM T58992 CU02RP 44405141 Ki > 5000 nM T58992 C1UZE3 44405145 Ki > 5000 nM T58992 CV5Y3I 44405172 Ki > 5000 nM T58992 CM05NC 44406109 Ki = 39 nM T58992 CA0RM2 44406110 Ki = 161 nM T58992 C2T6WY 44406111 Ki = 29 nM T58992 C5P9NO 44406128 Ki = 128 nM T58992 CI2C5K 44406161 Ki = 3696 nM T58992 CRL3P8 44406171 Ki = 29 nM T58992 CQ2D6B 44406177 Ki = 97 nM T58992 CALG92 44406185 Ki = 203 nM T58992 C7WQ5V 44406186 Ki = 217 nM T58992 CBH5G9 44406215 Ki = 3074 nM T58992 CRI8L5 44406219 Ki = 43 nM T58992 CUH65A 44406224 Ki = 31 nM T58992 CF61YM 44406225 Ki = 46 nM T58992 CKS9V8 44406273 Ki = 72 nM T58992 CS7KQ8 44406280 Ki > 465 nM T58992 CLE5R9 44406285 Ki = 9 nM T58992 CZFM30 44406286 Ki = 99 nM T58992 C57ADM 44406306 Ki = 44 nM T58992 CVX84Y 44406350 EC50 = 26 nM T58992 C0C2BN 44406353 Ki = 138 nM T58992 CJ6H4U 44406370 Ki = 46 nM T58992 C79UVP 44406376 Ki = 106 nM T58992 CZPS59 44406568 IC50 = 0.87 nM T58992 CL3EO9 44406605 IC50 = 260 nM T58992 C4RJY2 44406656 Ki = 700 nM T58992 CSMQ84 44406657 Ki = 8.3 nM T58992 CSF2Y6 44406658 Ki = 12 nM T58992 C2KBP7 44406663 Ki = 0.27 nM T58992 C3SEN7 44406695 Ki = 28 nM T58992 C2MR7W 44406696 Ki = 18 nM T58992 C4LA2U 44406703 Ki = 23 nM T58992 CZC51G 44406712 Ki = 38 nM T58992 CPO9T5 44406713 Ki = 160 nM T58992 CRE4Q9 44406723 Ki = 3.9 nM T58992 C4N1MC 44406724 Ki = 11 nM T58992 CB30EK 44406732 Ki = 4.4 nM T58992 CVER25 44407299 Ki = 680 nM T58992 C9AU3C 44407301 Ki = 120 nM T58992 CVP98E 44407305 Ki = 260 nM T58992 C4J3VF 44407309 Ki = 800 nM T58992 C3NG6O 44407310 Ki = 610 nM T58992 C7YM3D 44407311 Ki = 180 nM T58992 C2QNC5 44407312 Ki > 1000 nM T58992 C3DQ8W 44407313 Ki > 1000 nM T58992 CQ9X8L 44407315 Ki = 65 nM T58992 CX82DC 44407316 Ki = 320 nM T58992 CD9R7C 44407317 Ki > 1000 nM T58992 CY3EH0 44407318 Ki = 880 nM T58992 CU6D4P 44407323 Ki > 1000 nM T58992 CJ51HQ 44407324 Ki = 580 nM T58992 C2I8RZ 44407329 Ki > 1000 nM T58992 CW89MA 44407330 Ki > 1000 nM T58992 CTLY61 44407348 Ki = 710 nM T58992 CE9K1V 44407351 Ki > 1000 nM T58992 CY8R2X 44407359 Ki > 1000 nM T58992 C69OZA 44407360 Ki > 1000 nM T58992 CB16YW 44407361 Ki > 1000 nM T58992 C2P4ZH 44407364 Ki = 340 nM T58992 CD69PS 44408411 Ki = 0.48 nM T58992 C7QV6M 44408483 Ki = 3.4 nM T58992 C96ELC 44408632 Ki = 0.23 nM T58992 C59XVU 44411613 Ki > 10000 nM T58992 CYE4D3 44411762 Ki > 10000 nM T58992 CMG79P 44411790 Ki > 10000 nM T58992 CS0ZC2 44411794 Ki > 10000 nM T58992 CDK08M 44411860 Ki > 10000 nM T58992 C52WZH 44413231 Ki > 10000 nM T58992 CFJ64A 44413232 Ki > 5000 nM T58992 CNFC81 44413248 Ki > 5000 nM T58992 C0V4FI 44413286 Ki > 5000 nM T58992 CS7BI8 44413301 Ki > 5000 nM T58992 C1NGS0 44413314 Ki > 5000 nM T58992 C5J0BU 44413315 Ki > 5000 nM T58992 CH7E1C 44413329 Ki > 5000 nM T58992 C1OQ0L 44413330 Ki > 5000 nM T58992 CKV5S0 44413361 Ki > 5000 nM T58992 C5PHK7 44413362 Ki > 5000 nM T58992 CSQZ28 44413379 Ki > 5000 nM T58992 CCU2B5 44413384 Ki > 5000 nM T58992 CD5SZ9 44413385 Ki > 5000 nM T58992 C7GE2K 44413395 Ki > 5000 nM T58992 CCK6Y5 44413396 Ki > 5000 nM T58992 C0FL8K 44413401 Ki > 5000 nM T58992 C6J3HP 44413402 Ki > 5000 nM T58992 CB2OJ9 44413408 Ki > 5000 nM T58992 C82VJB 44413413 Ki > 5000 nM T58992 CP31JV 44413414 Ki > 5000 nM T58992 C98OQG 44413423 Ki > 5000 nM T58992 CH0DS7 44413441 Ki = 4180 nM T58992 CLSK72 44413442 Ki = 2750 nM T58992 CP75FM 44414890 Ki = 1.4 nM T58992 C3W9ZR 44415103 IC50 = 4895 nM T58992 C5XA2V 44415104 IC50 = 9048 nM T58992 C5DQU3 44415132 IC50 = 8260 nM T58992 CHA92Z 44415133 IC50 = 35616 nM T58992 CW97YG 44415143 IC50 = 10215 nM T58992 CPL8U5 44415144 IC50 = 56703 nM T58992 CSW4K9 44415190 IC50 = 8529 nM T58992 C7JI0K 44415191 IC50 = 10928 nM T58992 C1DH7S 44415192 IC50 = 17935 nM T58992 CNW4V0 44415202 IC50 = 48207 nM T58992 C3UC4M 44415224 IC50 = 3967 nM T58992 CNT96C 44415298 IC50 = 16984 nM T58992 C7EHS3 44415299 IC50 = 11273 nM T58992 C5Y7KT 44415300 IC50 = 10189 nM T58992 CCX92L 44415312 IC50 = 17799 nM T58992 C6EPF0 44415619 IC50 = 1.8 nM T58992 CU65WM 44415621 Ki = 110 nM T58992 C1MO6K 44415676 Ki = 9.9 nM T58992 C7U8LB 44415720 Ki = 210 nM T58992 C1UT9Q 44415832 Ki = 3.9 nM T58992 CDB98P 44416410 IC50 = 8400 nM T58992 C2LXG4 44416411 IC50 = 450 nM T58992 CPL16F 44416658 IC50 = 12100 nM T58992 C72RTL 44416659 IC50 = 6650 nM T58992 CZ4V9T 44416676 Ki = 7600 nM T58992 CUF36X 44417374 Ki = 0.63 nM T58992 CFJC63 44417384 Ki = 44.5 nM T58992 C5OI3W 44418923 Ki = 45 nM T58992 C4UPR1 44418924 Ki = 1.4 nM T58992 C72HIJ 44421393 Ki = 3.35 nM T58992 C0M1LF 44421396 Ki = 2.95 nM T58992 CI12ZC 44421399 Ki = 1.65 nM T58992 COM3F5 44421400 Ki = 1.81 nM T58992 C2L4MW 44421401 Ki = 2.94 nM T58992 CKA1J2 44421403 Ki = 3.1 nM T58992 C5S4EC 44421406 Ki = 1.8 nM T58992 CW6I0V 44421407 Ki = 1.63 nM T58992 CN6E4Q 44421408 Ki = 2.67 nM T58992 CLEH29 44421409 EC50 = 9.87 nM T58992 C4ZXO2 44421412 Ki = 4.17 nM T58992 C5K6YB 44421422 Ki = 5 nM T58992 C9ACE6 44422807 Ki = 28 nM T58992 C2IE1L 44422808 Ki = 15 nM T58992 C5OH7E 44423024 IC50 = 35100 nM T58992 CJPG01 44423028 IC50 = 86400 nM T58992 C4C3GM 44423035 IC50 = 32100 nM T58992 C0Q8TZ 44425152 Ki > 10000 nM T58992 C4NWJ9 44425154 Ki > 10000 nM T58992 CYQ28K 44425156 Ki > 10000 nM T58992 CN0P8A 44425365 Ki = 1700 nM T58992 C8N2JK 44425366 Ki = 260 nM T58992 C8Q6RA 44425367 Ki = 50 nM T58992 C5MV9B 44425368 Ki = 16000 nM T58992 CW01VE 44425369 Ki = 6900 nM T58992 CO14ZF 44425371 Ki = 76000 nM T58992 CK4ZI3 44425372 Ki = 15000 nM T58992 CWQ8Z3 44425373 Ki = 3300 nM T58992 CXO68V 44425374 Ki = 6500 nM T58992 C1JQ9U 44425375 Ki = 2400 nM T58992 CEH4T3 44425376 Ki = 2900 nM T58992 CV69GB 44425377 Ki = 9000 nM T58992 CE45JS 44425378 Ki = 12000 nM T58992 C5VUF4 44425379 Ki = 6300 nM T58992 C3J2RS 44425382 Ki = 15000 nM T58992 C10OMS 44426811 Ki = 348 nM T58992 C49KAS 44426813 Ki = 5323 nM T58992 CJ5FC0 44426816 Ki = 32960 nM T58992 C4TFP1 44426818 Ki = 121800 nM T58992 CP5V8D 44426821 Ki = 22295 nM T58992 C5L4SE 44426822 Ki = 21890 nM T58992 C36SCP 44426823 Ki = 10920 nM T58992 C72RXV 44426824 Ki = 7845 nM T58992 C0S5TE 44426829 Ki = 1271 nM T58992 CL1EG2 44426830 Ki = 7355 nM T58992 CBFY73 44426831 Ki = 10124 nM T58992 CFO9Q6 44426832 Ki = 237 nM T58992 C2NFA4 44426833 Ki = 3029 nM T58992 COJ48Z 44426834 Ki = 1431 nM T58992 CUD42S 44426835 Ki = 2945 nM T58992 CKJ90O 44426836 Ki = 2110 nM T58992 CZ4R6J 44426837 Ki = 4458 nM T58992 CPDE73 44426838 Ki = 1977 nM T58992 C53JGK 44426839 Ki > 100000 nM T58992 C7IJY0 44426840 Ki = 1783 nM T58992 CJB90W 44426841 Ki = 584 nM T58992 CK3B6E 44426843 Ki = 18160 nM T58992 CD3TB8 44426844 Ki = 13715 nM T58992 CFY3A6 44427433 Ki = 234 nM T58992 C0M4EP 44427434 Ki = 15 nM T58992 CF5OJ0 44430021 Ki = 28380 nM T58992 CUQ95Y 44430022 Ki = 4363 nM T58992 CZA0E6 44430023 Ki = 13905 nM T58992 CWX67P 44430033 Ki = 8885 nM T58992 C40BHT 44430038 Ki = 1212 nM T58992 C1QXR6 44430040 Ki = 2867 nM T58992 CS6Y5Z 44430042 Ki = 3702 nM T58992 C4CHV5 44430043 Ki = 3291 nM T58992 CX9P5R 44430044 Ki = 8435 nM T58992 CA51JN 44430045 Ki = 8900 nM T58992 C2G9HQ 44430046 Ki = 3990 nM T58992 C8PI4A 44430047 Ki = 9383 nM T58992 CL1N4D 44430048 Ki = 99505 nM T58992 C0AYM6 44430049 Ki = 23400 nM T58992 CMJT74 44430050 Ki = 3818 nM T58992 C4ZG6A 44430079 Ki = 1992 nM T58992 CSNQ43 44430080 Ki = 2445 nM T58992 CXV9J7 44430081 Ki = 2911 nM T58992 CFHY18 44430083 Ki = 1167 nM T58992 C6SBE1 44430084 Ki = 1705 nM T58992 CXZ2D3 44430085 Ki = 1585 nM T58992 CI4X3Z 44430087 Ki = 3159 nM T58992 C15KTO 44432560 Ki = 37 nM T58992 C47USK 44432561 Ki = 29 nM T58992 C9KQE6 44432562 Ki = 48 nM T58992 C8W2RQ 44432563 Ki = 23 nM T58992 CT4P1M 44432564 Ki = 37 nM T58992 CDP72X 44432565 Ki = 23 nM T58992 CJQC39 44432566 Ki = 125 nM T58992 CHNQ16 44432567 Ki = 29 nM T58992 C6TD1E 44432583 Ki = 85 nM T58992 CQ4X2F 44432589 Ki = 158 nM T58992 C97UQG 44432591 Ki = 19 nM T58992 CJN2O9 44432597 Ki = 9.3 nM T58992 CM3P1O 44432599 Ki = 7.4 nM T58992 C37YLC 44432606 Ki = 9.3 nM T58992 CA9S4M 44432608 Ki = 12 nM T58992 CG7KL2 44432609 Ki = 29 nM T58992 CLQH28 44432610 Ki = 12 nM T58992 C3W6AY 44432611 Ki = 5.9 nM T58992 CU8F0D 44432613 Ki = 51 nM T58992 CC15LP 44432614 Ki = 642 nM T58992 COM06U 44432615 Ki = 147 nM T58992 CG69US 44432616 Ki = 280 nM T58992 CF02PQ 44433159 Ki = 173 nM T58992 C34OTB 44433399 EC50 = 21 nM T58992 CT4QL9 44433400 Ki = 25 nM T58992 CO08LU 44433401 Ki = 110 nM T58992 CC5G2Y 44433402 EC50 = 57 nM T58992 CJ20NZ 44434062 Ki = 2351 nM T58992 CF78VR 44434063 Ki = 179.6 nM T58992 C38NOM 44434064 Ki = 2139 nM T58992 CT8QH4 44434065 Ki = 2448.94 nM T58992 CTM38X 44434066 Ki > 5000 nM T58992 CMT4U1 44434067 Ki = 169.39 nM T58992 CF0V8Z 44434068 Ki = 2708 nM T58992 C3H1NC 44434069 Ki = 1377 nM T58992 C39AJW 44434071 Ki = 503.7 nM T58992 C38LOE 44434072 Ki = 187 nM T58992 CR9GY1 44434075 Ki = 163.22 nM T58992 CT6ZD0 44434077 Ki = 232.46 nM T58992 COI7A6 44434079 Ki = 107.88 nM T58992 C73FSU 44434081 Ki = 239.77 nM T58992 CKEY87 44434082 Ki = 409.29 nM T58992 CLZ68X 44434084 Ki = 3888 nM T58992 CI2R7P 44434085 Ki = 388.15 nM T58992 C20PXC 44434087 Ki = 466.27 nM T58992 C1KB9R 44434088 Ki = 1909 nM T58992 CLU1X5 44434089 Ki = 2576 nM T58992 C72BXS 44434325 Ki = 73.8 nM T58992 C35HRS 44434326 Ki = 343.7 nM T58992 C0UK9Q 44434327 Ki = 77.7 nM T58992 C2CK7G 44434328 Ki = 208.5 nM T58992 C5J8VH 44434329 Ki = 269.4 nM T58992 C8CZX7 44434330 Ki = 93.1 nM T58992 C9DF1X 44434331 Ki = 698.1 nM T58992 C7CKX3 44434332 Ki = 59.6 nM T58992 CNFH86 44434333 Ki = 8.6 nM T58992 C5OW8M 44434334 Ki = 38.2 nM T58992 CS6BH9 44434335 Ki = 55.9 nM T58992 C61SUX 44434336 Ki = 5.3 nM T58992 CB2AQ4 44434932 Ki > 5000 nM T58992 C81KMS 44434933 Ki > 5000 nM T58992 COEG19 44434934 Ki > 5000 nM T58992 C9XW8Q 44434935 Ki > 5000 nM T58992 C4N9OY 44434936 Ki > 5000 nM T58992 C5UG8I 44434937 Ki > 5000 nM T58992 CGLY08 44434938 Ki = 214.73 nM T58992 C92WQA 44434939 Ki = 3458.36 nM T58992 C04LKG 44434940 Ki = 718.45 nM T58992 CT95NA 44434941 Ki = 673.58 nM T58992 CGKC17 44434942 Ki = 2414.41 nM T58992 CVF9O5 44434943 Ki > 5000 nM T58992 CUA32P 44434944 Ki = 128.07 nM T58992 CRBX46 44434945 Ki = 211.63 nM T58992 CD0R6I 44434947 Ki > 1000 nM T58992 CIN4E6 44434948 Ki > 1000 nM T58992 C2OCX5 44436083 Ki = 0.69 nM T58992 C87RIC 44436084 Ki = 0.36 nM T58992 CT30KJ 44437601 Ki = 1251 nM T58992 C1EHS4 44437602 Ki = 2123 nM T58992 CK73VO 44437606 Ki = 2020 nM T58992 CJ1ST3 44437610 Ki = 3411 nM T58992 C0M9SC 44437615 Ki = 3084 nM T58992 CTK2S0 44437619 Ki = 608 nM T58992 C4PK1O 44437623 Ki = 3084 nM T58992 CQKL94 44437636 Ki = 1471 nM T58992 C43URV 44437637 Ki = 1175 nM T58992 CRKH10 44437656 Ki = 320 nM T58992 CZB4Q9 44438912 Ki = 73655 nM T58992 C7RD2E 44438916 Ki = 8999 nM T58992 CNL30S 44438917 Ki = 724.5 nM T58992 C5D4NZ 44438920 Ki = 1035 nM T58992 CA2LD5 44438921 Ki = 6846 nM T58992 C6H7AD 44438922 Ki = 3373 nM T58992 CRN3W4 44438961 Ki = 1421 nM T58992 CGYD89 44438962 Ki = 736 nM T58992 CZ48KD 44438963 Ki = 11510 nM T58992 C2EGK7 44438964 Ki = 15715 nM T58992 COX57F 44438965 Ki = 14770 nM T58992 C9S2HB 44438966 Ki = 6042 nM T58992 C1HF6E 44438967 Ki = 24805 nM T58992 C3L7SB 44438968 Ki = 8600 nM T58992 CE63GK 44438971 Ki = 26515 nM T58992 C8TVI4 44438974 Ki = 16035 nM T58992 CPHS56 44438975 Ki = 10360 nM T58992 CK3Z5G 44438978 Ki = 5598 nM T58992 CPA4U5 44438983 Ki = 1231 nM T58992 C2TKY5 44438988 Ki = 2400 nM T58992 CL7WN5 44438993 Ki = 1375 nM T58992 C0A2OM 44439000 Ki = 1291 nM T58992 CMQA60 44439001 Ki = 2461 nM T58992 CH57IQ 44439874 Ki > 10000 nM T58992 CNS7T5 44439878 Ki > 10000 nM T58992 CF86GQ 44443051 Ki = 4.5 nM T58992 CHEI51 44443452 Ki = 5.1 nM T58992 CY78KN 44443453 Ki = 8.6 nM T58992 CF1IC2 44443454 Ki = 3.8 nM T58992 CDJ8T5 44444601 Ki = 0.18 nM T58992 C9N8VT 44444603 Ki = 2.5 nM T58992 C57TLG 44444604 Ki = 31 nM T58992 CBR38Y 44444613 Ki = 52 nM T58992 CT7M6Y 44447365 EC50 = 15.5 nM T58992 C56QDE 44448327 Ki = 6.2 nM T58992 CPW3J0 44448489 Ki = 4.4 nM T58992 CN9X6W 44448522 Ki = 23 nM T58992 C6TEA5 44448524 Ki = 0.85 nM T58992 CET3O5 44448563 Ki = 9.3 nM T58992 CJLI69 44450262 Ki = 11.8 nM T58992 C4NFQ9 44450499 Ki = 1410 nM T58992 CZ1R2D 44451649 Ki = 1288.25 nM T58992 C8KXY7 44452306 Ki = 740 nM T58992 CK1F5Z 44453675 Ki = 360 nM T58992 CRM8K4 44453699 Ki = 500 nM T58992 CUIC24 44453700 Ki = 10 nM T58992 C6QV3U 44453726 Ki = 15 nM T58992 C5HM3F 44453728 Ki = 3.2 nM T58992 CDY56P 44453750 Ki = 31 nM T58992 CO56PJ 44453779 Ki = 8.3 nM T58992 CO2XU7 44453801 Ki = 74 nM T58992 COI2B9 44453822 Ki = 22 nM T58992 CR1S3K 44453824 Ki = 24 nM T58992 C4ID6Y 44453825 Ki = 52 nM T58992 CBUE46 44453848 Ki = 63 nM T58992 CZ7X2D 44453849 Ki = 39 nM T58992 CTEK70 44453879 Ki = 67 nM T58992 CH1D0B 44453880 Ki = 29 nM T58992 CA05FK 44453881 Ki = 100 nM T58992 CTO26R 44453900 Ki = 620 nM T58992 CN7B2P 44453901 Ki = 360 nM T58992 C1PQA7 44453924 Ki = 170 nM T58992 C81IOK 44453925 Ki = 160 nM T58992 C12XGE 44456400 Ki > 10000 nM T58992 C9KU1O 44456785 Ki = 8.22 nM T58992 C6PEF7 44456833 Ki = 8.5 nM T58992 C3V7WR 44457580 Ki = 2650 nM T58992 C4SQ7V 44457667 Ki = 39.5 nM T58992 CJ3KG5 44457676 Ki = 317 nM T58992 C2I8RC 44458295 IC50 > 10000 nM T58992 CVM72Y 44458341 IC50 > 10000 nM T58992 CQ0WM7 44469273 IC50 > 5000 nM T58992 C0N2XB 44474938 Ki = 209 nM T58992 CL5NO6 44541248 Ki = 3.26 nM T58992 C6K3GX 44541249 Ki = 1.6 nM T58992 CVX16Z 44541250 Ki = 28.3 nM T58992 C29MSC 44541387 Ki = 65.2 nM T58992 CI9O3F 44541388 Ki = 5.41 nM T58992 C6TW8L 44541389 Ki = 136 nM T58992 C6T1UX 44551464 Ki = 1.4 nM T58992 CQKE48 44564372 Ki = 1441 nM T58992 CRX6D7 44568828 Ki = 500 nM T58992 CMT15I 44568829 Ki = 160 nM T58992 CL80WF 44570025 Ki = 220 nM T58992 C9ERN6 44570030 Ki > 10000 nM T58992 CP2M8D 44570031 Ki = 54 nM T58992 CN7UA9 44570032 Ki = 1000 nM T58992 CPA48R 44570066 Ki = 320 nM T58992 CGK40O 44570070 Ki = 14 nM T58992 C6C0XR 44570071 Ki = 1000 nM T58992 CT10RB 44570072 Ki > 10000 nM T58992 C8P3SX 44570073 Ki = 67 nM T58992 CB01RQ 44570075 Ki > 10000 nM T58992 CO4NI2 44573249 EC50 = 5 nM T58992 C9OF8P 44573250 EC50 = 24 nM T58992 CPJ27Z 44573251 EC50 = 13 nM T58992 CIK5T2 44573291 EC50 = 83 nM T58992 CM89KA 44573292 EC50 = 14 nM T58992 CI6F0Y 44573293 EC50 = 59 nM T58992 CL6C7B 44573294 EC50 = 60 nM T58992 CBM82T 44573332 EC50 = 171 nM T58992 CP6GE8 44573333 EC50 = 207 nM T58992 CT5SY1 44573334 EC50 = 308 nM T58992 CMSV07 44573403 EC50 = 846 nM T58992 CLX14F 44573404 EC50 = 30 nM T58992 C0PD8L 44573405 EC50 = 52 nM T58992 CA03TK 44573444 EC50 = 108 nM T58992 CZ26TO 44573445 EC50 = 3 nM T58992 CQ9WA5 44573446 EC50 = 28 nM T58992 CKJ2O8 44573447 EC50 = 41 nM T58992 C4ZCX6 44576628 EC50 = 14 nM T58992 C8HF3V 44577045 Ki > 10000 nM T58992 CRME18 44577046 Ki = 220 nM T58992 CI1L7Y 44577047 Ki = 730 nM T58992 CDPS18 44577048 Ki = 35 nM T58992 C8OU4Q 44577049 Ki = 2000 nM T58992 CGMC75 44577468 Ki = 120 nM T58992 CZUW31 44577469 Ki > 10000 nM T58992 CES86D 44577470 Ki = 52 nM T58992 CU6ZT4 44577524 Ki = 1500 nM T58992 CXS42P 44577525 Ki = 410 nM T58992 CWIG26 44577526 Ki = 1000 nM T58992 CTIH86 44577527 Ki = 1900 nM T58992 CDT46S 44578135 Ki = 40 nM T58992 CRK51Y 44581834 Ki > 10000 nM T58992 CG1DL2 44582176 Ki = 1441 nM T58992 C3YMV4 44582184 Ki = 170.3 nM T58992 CKFX03 44582185 Ki = 405.32 nM T58992 CK8G4D 44582186 Ki > 10000 nM T58992 CIX09B 44582198 Ki > 10000 nM T58992 CC06XI 44582199 Ki = 22.81 nM T58992 CEUS82 44582200 Ki = 818.43 nM T58992 C28VHY 44582218 Ki = 907.18 nM T58992 CM21UD 44583389 Ki > 1000 nM T58992 C6YOC5 44583390 Ki > 1000 nM T58992 CX1L5P 44583391 Ki > 1000 nM T58992 C7PCJ1 44583392 Ki > 1000 nM T58992 CAHK35 44583425 Ki > 1000 nM T58992 C7VWA3 44583426 Ki > 1000 nM T58992 CNG34J 44583429 Ki > 1000 nM T58992 CHZ46N 44583430 Ki > 1000 nM T58992 CASI92 44583431 Ki > 1000 nM T58992 CLAR69 44583432 Ki > 1000 nM T58992 CJOH07 44586888 Ki = 12 nM T58992 CJS8F2 44586890 Ki = 190 nM T58992 CP2N8S 44586914 Ki = 63 nM T58992 C7P0XN 44586916 Ki = 96 nM T58992 CV9H6N 44586918 Ki = 22 nM T58992 CP8EX5 44586920 Ki = 690 nM T58992 C1I0RO 44586943 Ki = 23 nM T58992 C5KN8O 44586945 Ki = 760 nM T58992 CZ9NA4 44586947 Ki = 490 nM T58992 CH97QC 44586949 Ki = 670 nM T58992 C8A9WK 44586979 Ki = 500 nM T58992 CZ28KA 44586981 Ki = 1500 nM T58992 CYC3Z6 44586983 Ki = 930 nM T58992 C1HA0F 44588005 Ki = 3430 nM T58992 CS1G0I 44588006 Ki = 2840 nM T58992 CT3C8S 44588007 Ki = 2530 nM T58992 CDMZ71 44588493 Ki > 10000 nM T58992 CVCW78 44588494 Ki = 4760 nM T58992 CN7OR6 44588495 Ki = 10000 nM T58992 CZIM85 44588496 Ki = 3710 nM T58992 C6EQ3R 44590514 IC50 = 7161 nM T58992 CEXW79 44590551 IC50 = 3795 nM T58992 C5UIT4 44590552 IC50 = 1274 nM T58992 CP83ZW 44590553 IC50 = 3947 nM T58992 C1AP0B 44590554 IC50 = 3620 nM T58992 C4U3AE 44590580 IC50 = 3887 nM T58992 CBS8P1 44590581 IC50 = 1467 nM T58992 C41SFR 44590582 IC50 = 1955 nM T58992 CD70YK 44590629 IC50 = 2289 nM T58992 CY36KS 44590630 IC50 = 1243 nM T58992 C60XNA 44590631 IC50 > 10000 nM T58992 CJ3R7Q 44590632 IC50 = 3501 nM T58992 CMH26K 44590677 IC50 > 10000 nM T58992 CN8S5P 44590678 IC50 > 10000 nM T58992 CFLP28 44591164 Ki = 5.1 nM T58992 C8ZC6O 44591193 Ki = 18 nM T58992 CEA9O2 44591194 Ki = 730 nM T58992 CER74Z 44591195 Ki = 51 nM T58992 CIU9T1 44591196 Ki = 680 nM T58992 CO3P8X 44591197 Ki = 160 nM T58992 CN5ZF8 44591198 Ki = 46 nM T58992 CZJ16A 44591987 Ki = 150 nM T58992 C6A1PL 44592015 EC50 = 3.7 nM T58992 CB3VG2 44592016 Ki = 280 nM T58992 CXL41O 44592053 Ki = 78 nM T58992 C3VSJ2 44592054 Ki > 10000 nM T58992 CNI1E9 44592056 Ki = 900 nM T58992 CUW6Q3 44592086 Ki = 4.2 nM T58992 C8DS7Q 44592087 Ki = 630 nM T58992 CU5GE1 44592088 Ki = 8.3 nM T58992 C9GRS1 44592089 Ki = 260 nM T58992 CPX7G6 44592124 Ki = 0.3 nM T58992 CDPU87 44596170 EC50 = 0.2 nM T58992 C2EC4H 44597424 Ki = 2490 nM T58992 CJ69LZ 44597425 Ki = 3100 nM T58992 C3ASC5 44597529 Ki = 443 nM T58992 C6XHL0 44597530 Ki = 807 nM T58992 CAOX39 44597597 Ki = 37 nM T58992 C2C9LF 44597714 Ki = 15 nM T58992 CEOB85 44597715 Ki = 50 nM T58992 C1R3QC 44597828 Ki = 42 nM T58992 CRS74M 44597830 Ki = 210 nM T58992 C39PTC 44597831 Ki = 20 nM T58992 C14EJV 44597940 Ki = 390 nM T58992 C3Q0ZL 44601476 IC50 > 32000 nM T58992 CVH94R 44608034 IC50 > 32000 nM T58992 CH68PJ 44620907 IC50 > 32000 nM T58992 C3DCT2 44626536 Ki = 94 nM T58992 CUZY73 44626538 Ki = 250 nM T58992 CG8W0U 44626542 Ki > 10000 nM T58992 CY6D4O 44626643 Ki > 10000 nM T58992 CB9JD0 44626647 Ki > 10000 nM T58992 C25QXW 44626747 Ki > 10000 nM T58992 C2NC5S 44626748 Ki = 190 nM T58992 C6GB5A 44626749 Ki = 850 nM T58992 CCZ89E 44626842 Ki = 1000 nM T58992 CKRL83 44627034 Ki = 1100 nM T58992 CBNJ20 44627035 Ki = 710 nM T58992 CVD03Q 44627135 Ki = 1600 nM T58992 C8XG3W 44627136 Ki = 730 nM T58992 C8PK2F 44627248 Ki = 72 nM T58992 C81KJQ 44627363 Ki = 610 nM T58992 C8NJR1 44627679 Ki > 10000 nM T58992 C7CJM9 44627680 Ki = 34 nM T58992 CM49FS 44627786 Ki = 190 nM T58992 C81LTN 44627787 Ki = 20 nM T58992 CPTL91 44627788 Ki = 120 nM T58992 CZ6VP4 44627789 Ki = 960 nM T58992 CQZ0W4 44627899 Ki = 1.7 nM T58992 C6AR0U 44627902 Ki = 19 nM T58992 CK0T4Y 44627998 Ki = 14.6 nM T58992 C79JNE 44627999 Ki = 67 nM T58992 CVI57S 44628102 Ki = 16 nM T58992 CS8X1U 44665679 IC50 > 32000 nM T58992 CR3PL6 44665680 IC50 > 32000 nM T58992 CT5CK8 44665687 IC50 > 32000 nM T58992 C3HXK5 45100475 IC50 > 32000 nM T58992 C45PUQ 45102745 Ki = 7000 nM T58992 C4LOY2 45115589 IC50 > 32000 nM T58992 CU8I6T 45263517 Ki = 503 nM T58992 CVDQ53 45265789 Ki = 8765 nM T58992 C40CHQ 45269407 Ki = 334 nM T58992 CT1U4X 45270231 Ki = 74.6 nM T58992 C7HF9D 45271055 Ki = 93.1 nM T58992 C6FEH0 45271306 Ki = 0.77 nM T58992 C7ZWN3 45272750 Ki = 0.12 nM T58992 C05BPC 45273694 Ki = 0.83 nM T58992 CIL49C 45482634 Ki = 5.1 nM T58992 CAP40I 45483185 Ki = 34.3 nM T58992 CMN6O9 45483211 Ki = 3.4 nM T58992 CFR5M7 45483251 Ki = 80.6 nM T58992 CL7KU2 45483259 Ki = 1.7 nM T58992 C8DOR2 45483260 Ki = 447 nM T58992 CFU8K5 45483286 Ki = 11.7 nM T58992 CHN46U 45483287 Ki = 435 nM T58992 C1X8JY 45483646 Ki = 38.1 nM T58992 CGOZ34 45483648 Ki = 60.3 nM T58992 CI8M5T 45483656 Ki = 19.4 nM T58992 CI6BL3 45483657 Ki = 110 nM T58992 CE13WZ 45483658 Ki = 2.01 nM T58992 CEZJ19 45483659 Ki = 32 nM T58992 C43JND 45483664 Ki = 0.41 nM T58992 C49WAV 45483668 Ki = 1.37 nM T58992 CVC0G3 45483672 Ki = 1.79 nM T58992 C0J4CG 45483978 Ki = 39 nM T58992 CFY46C 45483979 Ki = 130 nM T58992 CC69WR 45483986 IC50 = 23.8 nM T58992 CLMP13 45483987 IC50 = 342 nM T58992 C3TJ9O 45483988 IC50 = 272 nM T58992 CPO50D 45483989 IC50 = 97.1 nM T58992 CQ5G8V 45483990 IC50 = 382 nM T58992 CKB8H3 45483991 IC50 = 436 nM T58992 C89UEA 45485826 Ki = 0.99 nM T58992 C76IZT 45485837 Ki = 49.6 nM T58992 C2DRY1 45485876 Ki = 18.2 nM T58992 CBW8D7 45485877 Ki = 11.1 nM T58992 C2OE9C 45485974 Ki = 50.2 nM T58992 CBP10O 45485982 Ki = 14 nM T58992 CS2IC5 45485986 Ki = 22.8 nM T58992 CGB37Y 45486011 Ki = 0.76 nM T58992 C1TJC6 45486012 Ki = 1.02 nM T58992 CHQI57 45486013 Ki = 1.7 nM T58992 C0KXD9 45486018 Ki = 0.24 nM T58992 CF46MY 45486027 Ki = 1.03 nM T58992 C9DVC1 45486028 Ki = 2.3 nM T58992 C3EV6H 45486032 Ki = 0.97 nM T58992 CV1N7L 45486033 Ki = 1.61 nM T58992 C9F4WP 45486035 Ki = 0.7 nM T58992 CC6DZ4 45486042 EC50 = 0.22 nM T58992 CE1MR2 45486046 EC50 = 0.22 nM T58992 CW7I8C 45486055 Ki = 0.42 nM T58992 C5JE6L 45486062 Ki = 1.4 nM T58992 CL2QF9 45486070 Ki = 0.42 nM T58992 CM39DL 45486096 Ki = 0.65 nM T58992 C60VCS 45486101 Ki = 0.64 nM T58992 CGY05X 45486102 Ki = 0.3 nM T58992 C6YS7G 45486258 Ki = 610 nM T58992 C8CKM0 45487174 Ki = 6 nM T58992 CSC23N 45487200 Ki = 544 nM T58992 CFC45O 45487206 Ki = 490 nM T58992 C3QU2C 45487384 IC50 > 5000 nM T58992 CO7VJ6 46190938 Ki = 2 nM T58992 CO0Z6H 46190939 Ki = 7 nM T58992 CV89LB 46226159 Ki = 1.8 nM T58992 COZ08F 46226176 Ki = 2.3 nM T58992 CL10HJ 46226250 Ki = 39 nM T58992 CZ5T6V 46227360 Ki = 5 nM T58992 CWC4L2 46227361 Ki = 7.8 nM T58992 CZ61KI 46227362 EC50 = 0.01738 nM T58992 C37HPA 46227363 EC50 = 13 nM T58992 C3YHF0 46227961 Ki = 0.1 nM T58992 C7LW1S 46227963 Ki = 2.5 nM T58992 C9L6WI 46227966 EC50 = 0.3 nM T58992 C6RK5N 46230439 Ki > 4300 nM T58992 CSD7C9 46230440 Ki = 7480 nM T58992 CK4TO1 46230441 Ki = 7210 nM T58992 C7L1QA 46230532 Ki = 2260 nM T58992 C5UZ4O 46230533 Ki = 6150 nM T58992 C2QE0Y 46230534 Ki > 4500 nM T58992 CDF6P8 46230535 Ki > 4500 nM T58992 CC85FR 46237455 Ki > 1000 nM T58992 CMJ0K7 46237580 Ki > 1000 nM T58992 C3R4KL 46237583 Ki > 1000 nM T58992 CC0K6V 46237584 Ki > 1000 nM T58992 CSH53K 46237585 Ki > 1000 nM T58992 CQ6K9E 46237703 Ki > 1000 nM T58992 C0G6MX 46237708 Ki > 1000 nM T58992 CNC81F 46237832 Ki > 1000 nM T58992 C97MLP 46237834 Ki > 1000 nM T58992 C45EPA 46237835 Ki > 1000 nM T58992 CAY07H 46237836 Ki > 1000 nM T58992 CCP98G 46237837 Ki > 1000 nM T58992 CPNX59 46782151 Ki = 1690 nM T58992 CKDW26 46831098 Ki > 10000 nM T58992 C5V6JT 46831100 Ki = 7300 nM T58992 CK4D7I 46865103 Ki > 200000 nM T58992 C6EX2B 46865104 Ki > 200000 nM T58992 C8OK1P 46867404 EC50 = 380 nM T58992 C0J5XV 46867466 Ki = 187 nM T58992 C9NGO7 46869046 IC50 = 2.7 nM T58992 CO5NQ3 46877612 Ki = 1.9 nM T58992 CDQ38I 46877614 Ki = 10 nM T58992 C0KM4A 46877617 Ki = 77 nM T58992 CFT10Y 46877619 Ki = 2.4 nM T58992 CW0J3V 46877621 Ki = 0.6 nM T58992 CI05BR 46877624 Ki = 0.14 nM T58992 C2CQF8 46877629 Ki = 0.02 nM T58992 CF9G0A 46877633 Ki = 0.407 nM T58992 C50ACR 46877637 Ki = 5.5 nM T58992 C0C5SR 46877643 Ki = 0.9 nM T58992 CQ26HB 46877644 Ki = 0.99 nM T58992 CVU37F 46877653 Ki = 2.57 nM T58992 CG19YU 46877660 Ki = 36.8 nM T58992 CWF58D 46877669 Ki = 0.96 nM T58992 CWT3O2 46877673 Ki = 0.12 nM T58992 CY8TW9 46877674 Ki = 15 nM T58992 CC40AZ 46877676 Ki = 7.8 nM T58992 C1V9KZ 46877677 Ki = 1.5 nM T58992 CM24KW 46877761 IC50 = 5.3 nM T58992 CK0G5J 46877762 IC50 = 450 nM T58992 CWX34Z 46877763 IC50 = 240 nM T58992 C2APF6 46877765 IC50 = 22 nM T58992 CQ4XP2 46877816 Ki = 1.1 nM T58992 CS53GL 46877852 Ki = 163 nM T58992 CUN8X2 46877853 Ki = 25.5 nM T58992 CAY0L4 46877854 Ki = 50.6 nM T58992 CZG2E3 46877855 Ki = 181 nM T58992 C3K6HF 46877888 Ki = 3500 nM T58992 CK7CY0 46878243 Ki = 4 nM T58992 CUMN01 46878245 Ki = 0.54 nM T58992 CJR0C1 46878247 Ki = 1.25 nM T58992 C4LCV8 46880270 Ki = 94000 nM T58992 C8T5GF 46880271 Ki > 200000 nM T58992 CWK29B 46880272 Ki > 200000 nM T58992 C7HT9Q 46880391 Ki = 180 nM T58992 CARP46 46880392 Ki = 37 nM T58992 C12DCB 46880393 Ki = 33 nM T58992 C65ALC 46880394 Ki = 420 nM T58992 CKQ94Y 46880395 Ki = 160 nM T58992 C5HDU1 46880396 Ki = 74 nM T58992 C82AOZ 46880397 Ki = 99 nM T58992 CW3F8K 46880398 Ki = 27 nM T58992 CKJD61 46880399 Ki = 29 nM T58992 C1RZ7T 46880400 Ki = 200 nM T58992 CV7K6J 46880401 Ki = 52 nM T58992 C49NWA 46880452 Ki = 20 nM T58992 C7JK5C 46880453 Ki = 920 nM T58992 CE6Y5T 46880454 Ki = 86 nM T58992 C0YJ1U 46928474 Ki = 750 nM T58992 CQ86RS 46928475 Ki = 43 nM T58992 C0HQ9F 46928476 Ki = 740 nM T58992 CI86QW 46928478 Ki = 25 nM T58992 CR3O7S 46928581 Ki = 1100 nM T58992 CV93BN 46945445 Ki > 10000 nM T58992 C0H1AC 46945446 Ki > 10000 nM T58992 CABL63 49765080 IC50 > 30000 nM T58992 C2LZJ0 49783209 Ki > 10000 nM T58992 C57SMG 49783415 Ki > 10000 nM T58992 C0TG6I 49783419 Ki > 10000 nM T58992 C8Y2QS 49798104 Ki = 2300 nM T58992 C6LEM8 49798106 Ki = 1300 nM T58992 C8EG6Y 49798111 Ki = 6.2 nM T58992 C24DUW 49798112 Ki = 2.9 nM T58992 COJG46 49799947 IC50 = 4.1 nM T58992 CYP36E 49799951 Ki > 1000 nM T58992 CTR1Y2 49799964 Ki = 1.1 nM T58992 CDS18H 49799966 Ki = 77.5 nM T58992 C4FA1V 49799967 Ki = 12.9 nM T58992 CEG52T 49799968 Ki = 7 nM T58992 C2H8LY 49799969 Ki = 0.7 nM T58992 C3T6NH 49843555 Ki > 5000 nM T58992 C9M7FZ 49863731 Ki = 1.7 nM T58992 C9PCU7 49863732 Ki = 38 nM T58992 C92LUS 49863733 Ki = 150 nM T58992 C97UJR 49863734 EC50 = 120 nM T58992 CU18KV 49863750 Ki = 16 nM T58992 CXW97O 49865703 IC50 > 30000 nM T58992 CRG60N 49865732 IC50 > 30000 nM T58992 CZY2T3 49865733 IC50 = 27442 nM T58992 CI2W0D 49865783 IC50 = 24290 nM T58992 CUK35O 49865784 IC50 > 30000 nM T58992 CLD4P0 49865785 IC50 > 30000 nM T58992 CL0DR3 49865859 IC50 = 14697 nM T58992 C2RY0J 50878551 Ki > 10000 nM T58992 C1W6TV 50898777 Ki > 10000 nM T58992 CXMZ73 50898778 Ki > 10000 nM T58992 C9W0VY 50925450 Ki = 0.14 nM T58992 CG4SX0 50942591 Ki > 10000 nM T58992 CWH2U8 50994380 EC50 = 0.1 nM T58992 CXIE93 50994381 Ki = 1.1 nM T58992 C9WUA6 50994458 Ki = 1.7 nM T58992 CIB51C 50994459 EC50 = 0.06457 nM T58992 C2GM0W 50994460 EC50 = 0.07 nM T58992 CIOV03 50994461 Ki = 19 nM T58992 CU63SQ 50994498 Ki > 1000 nM T58992 CWA5D8 50994529 Ki = 1.6 nM T58992 C09NJQ 50994530 Ki = 0.03 nM T58992 CEDJ62 50994531 EC50 = 0.08511 nM T58992 C0Y5GB 50994602 Ki = 0.11 nM T58992 C5D0NY 51002736 Ki = 152 nM T58992 C3OQP7 51002739 Ki = 359 nM T58992 CBPQ82 51002822 Ki = 200 nM T58992 CCTI18 51002823 Ki = 165 nM T58992 CFGZ31 51002824 Ki = 196 nM T58992 CSW52C 51002825 Ki = 1980 nM T58992 C8OFC7 51002870 Ki = 138 nM T58992 CG7US6 51002874 Ki = 454 nM T58992 C0B8ZH 51002978 Ki = 183 nM T58992 C7FI2R 51002981 Ki = 800 nM T58992 C7QA4S 51003039 Ki = 547 nM T58992 CGU3H2 51003042 Ki = 610 nM T58992 C08HUZ 51003216 EC50 = 1.06 nM T58992 CXW86B 51003218 EC50 = 0.69 nM T58992 CW5Q7V 51003448 Ki = 158.49 nM T58992 CGR98N 51003449 Ki = 12.59 nM T58992 C9WEO3 51003467 Ki = 0.58 nM T58992 CNV2Q4 51004758 IC50 > 10000 nM T58992 C1SK7C 51009928 IC50 > 10000 nM T58992 CM2K7S 51042171 Ki = 5.7 nM T58992 CE4KP1 51050257 Ki > 10000 nM T58992 CQ6SR3 51353734 Ki = 91 nM T58992 CDQ3I6 51353736 Ki = 50 nM T58992 C4GH6F 51353738 Ki = 120 nM T58992 CZ1CL5 51353740 Ki = 420 nM T58992 C3W7AJ 51353742 Ki = 220 nM T58992 CK07VQ 51353744 Ki = 76 nM T58992 C9JAE4 51356293 Ki = 54 nM T58992 C7MNL4 51356294 Ki = 56 nM T58992 C3S0LD 51356295 Ki = 180 nM T58992 C6OY1E 51356296 Ki = 34 nM T58992 C54EPI 51356297 Ki = 41 nM T58992 CAU84H 51356590 Ki = 29 nM T58992 CZ1GB9 51356591 Ki = 150 nM T58992 CE16YQ 51356593 Ki = 140 nM T58992 CGF0L6 51356594 Ki > 10000 nM T58992 CY5A7R 51357141 Ki = 47 nM T58992 CQ5Y6C 51357143 Ki = 79 nM T58992 CYB1A0 51357420 Ki = 65 nM T58992 C2VN8I 52937468 Ki = 0.6 nM T58992 C1M3SD 52941462 IC50 = 2145 nM T58992 CPOQ82 52942580 IC50 > 30000 nM T58992 C3YF5D 52942581 IC50 > 30000 nM T58992 C5V4DW 52943162 IC50 = 10914 nM T58992 CNK14O 52943803 IC50 = 4842 nM T58992 C89GIK 52944552 IC50 > 21889 nM T58992 CV48KS 52945118 IC50 = 2668 nM T58992 CWA1T5 52945160 IC50 = 12 nM T58992 CSZ4R3 52945588 IC50 = 4000 nM T58992 CNGU78 52945626 IC50 = 11076 nM T58992 CG8CN4 52946340 IC50 > 30000 nM T58992 C41AYU 52947523 IC50 > 27287 nM T58992 CFI96N 52947735 IC50 > 30000 nM T58992 CI63UL 52948240 IC50 > 24727 nM T58992 CAID24 52948615 IC50 > 30000 nM T58992 C48RBH 52948719 IC50 > 30000 nM T58992 CZX5B9 52948735 IC50 = 5389 nM T58992 CVWY23 52949439 IC50 = 22049 nM T58992 C01KMG 52952006 Ki = 2260 nM T58992 CL1QG4 52952007 Ki > 5000 nM T58992 CET8Q0 52952008 Ki > 10000 nM T58992 C6X7WL 52952107 Ki > 5200 nM T58992 C4N9HF 52952108 Ki > 5000 nM T58992 CWC1N8 52952109 Ki > 5000 nM T58992 C7JB4Q 52952110 Ki > 5000 nM T58992 C2GPE5 52952207 Ki > 5000 nM T58992 CTU43X 53316968 Ki > 500 nM T58992 CCOD69 53316969 Ki > 5000 nM T58992 CE3P7Y 53317205 Ki = 251.19 nM T58992 C0NKY7 53317262 Ki = 63.1 nM T58992 C7H8QK 53318490 Ki = 1584.89 nM T58992 C31ZOA 53318757 Ki = 501.19 nM T58992 CI6CQ0 53319615 Ki = 205 nM T58992 C6SY4G 53319616 Ki = 312 nM T58992 CB10OV 53319822 Ki = 39.81 nM T58992 CT8R3I 53319870 Ki = 316.23 nM T58992 C4XD5Q 53319871 Ki = 100 nM T58992 CY5MG9 53321111 Ki > 3981.07 nM T58992 CD14AE 53321176 Ki > 3981.07 nM T58992 C6X9OT 53321653 Ki > 3981.07 nM T58992 C2EV1S 53322245 Ki > 500 nM T58992 CRN26Z 53322438 Ki = 398.11 nM T58992 CZY2G3 53322439 Ki = 316.23 nM T58992 CMOL62 53322496 Ki = 100 nM T58992 CLDI90 53323074 Ki = 1.6 nM T58992 C30TBO 53323800 Ki = 251.19 nM T58992 CS9I6Z 53323801 Ki = 398.11 nM T58992 CGI94L 53323802 Ki = 79.43 nM T58992 C5I4KQ 53323803 Ki = 316.23 nM T58992 C0ZJ1T 53323804 Ki = 158.49 nM T58992 CV5EC1 53323805 Ki = 100 nM T58992 C7Z4KR 53323841 Ki > 3981.07 nM T58992 C32YWL 53324045 Ki = 1526 nM T58992 C9YF7G 53324694 Ki = 4.2 nM T58992 CJ59GU 53325079 Ki = 50.12 nM T58992 CH37ZT 53325227 Ki > 10000 nM T58992 CRQF15 53325242 Ki = 1413 nM T58992 C5E7LW 53325608 Ki = 679 nM T58992 CL5WG8 53325725 IC50 = 0.81 nM T58992 CRZ76L 53326167 Ki = 258 nM T58992 CLP1Q0 53326367 Ki = 316.23 nM T58992 C7ETI8 53326368 Ki = 199.53 nM T58992 CL7I4V 53326806 Ki = 105 nM T58992 CI3K7N 53326835 Ki = 316.23 nM T58992 CA3KL4 53388149 EC50 = 38.6 nM T58992 C0TIQ5 53388316 EC50 = 19 nM T58992 CZ2M7C 53388784 IC50 = 5400 nM T58992 C70BZV 54580938 Ki = 8 nM T58992 CYEC84 54581367 Ki > 10000 nM T58992 CUH4E9 54581461 Ki = 0.15 nM T58992 C3I0HF 54582933 Ki = 35 nM T58992 C9G8RT 54582934 Ki = 170 nM T58992 CX0O1G 54583374 Ki = 190 nM T58992 CHA7T8 54584041 Ki = 14 nM T58992 C96ISF 54584882 Ki = 8.1 nM T58992 CKUH91 54585844 Ki = 39 nM T58992 C6MHV9 54585845 Ki = 39 nM T58992 CV86NQ 54586810 Ki = 13 nM T58992 C3EP9X 54669894 EC50 = 0.016 nM T58992 C50VRZ 54678117 Ki = 2 nM T58992 C0IT4S 54678127 Ki = 7.4 nM T58992 CQIS61 54678129 Ki = 16 nM T58992 CH1LY5 54678130 Ki = 6.8 nM T58992 CGVW28 54718272 Ki = 11.1 nM T58992 CXF1G9 54751920 Ki > 100000 nM T58992 CNT03F 54754507 Ki = 24 nM T58992 CROS84 54756989 Ki = 1.27 nM T58992 C2ISE6 54756990 Ki = 3.66 nM T58992 C7F6EC 54757387 EC50 = 0.17 nM T58992 CQU87I 56589659 EC50 = 1.1 nM T58992 CHZ1D7 56589680 EC50 = 11 nM T58992 C28AED 56655502 Ki = 211 nM T58992 CCN2E8 56658044 Ki = 7.13 nM T58992 CJW5C1 56658452 Ki = 502.4 nM T58992 C69VIF 56661555 Ki = 17.2 nM T58992 CJ2MA7 56663008 Ki = 2.55 nM T58992 CUE0R7 56664847 IC50 = 3.4 nM T58992 CDKP63 56664973 Ki = 1.59 nM T58992 CEW3K4 56665405 Ki = 294 nM T58992 CR64WX 56665407 Ki = 865.6 nM T58992 C3QLV1 56666529 Ki > 5000 nM T58992 C4QM3N 56668405 Ki = 6.79 nM T58992 C8O7MT 56668839 Ki = 602.2 nM T58992 CL21RS 56669900 Ki = 70.76 nM T58992 CO18SG 56669938 Ki > 4900 nM T58992 C9SY1A 56672310 Ki = 90.1 nM T58992 C9Y4VR 56674946 Ki = 50 nM T58992 CD9JK4 56675713 Ki = 128 nM T58992 C45KMW 56676759 Ki > 4900 nM T58992 C0WVZ6 56676760 Ki > 4900 nM T58992 CVXJ29 56676761 Ki > 4900 nM T58992 C7EFI9 56678759 IC50 = 17.4 nM T58992 CQZ75Y 56678873 Ki = 1250 nM T58992 CZ6B0O 56678874 Ki = 1230 nM T58992 C15FOK 56679008 Ki = 173.7 nM T58992 CDG30L 56680069 Ki > 5000 nM T58992 CX8F2N 56681954 Ki = 3.03 nM T58992 C2A4MQ 56681955 Ki = 8.67 nM T58992 CK52GV 56682330 Ki = 2586 nM T58992 C95LAM 56834761 Ki = 130 nM T58992 CRX31L 56840667 Ki = 152 nM T58992 CQ2O4U 56849549 Ki > 500 nM T58992 CCMS01 56849550 Ki > 500 nM T58992 C7VT5K 56849551 Ki > 500 nM T58992 C2Y9CE 56851423 Ki > 500 nM T58992 C34PMD 56851424 Ki > 500 nM T58992 CN32ZB 56851582 Ki = 251 nM T58992 CY9DH2 56851583 Ki = 153 nM T58992 CC3JS8 56851584 Ki > 500 nM T58992 C9E6CU 56851585 Ki > 500 nM T58992 C1ZOM5 56851586 Ki = 165 nM T58992 CSH7D9 57390216 IC50 = 0.071 nM T58992 CLN2F8 57390217 IC50 = 4.1 nM T58992 CAF23D 57390707 EC50 = 2.34 nM T58992 CS1K0A 57391716 Ki = 1000 nM T58992 CZ1EH9 57391826 IC50 = 2.4 nM T58992 C3MUQ4 57392006 IC50 = 0.27 nM T58992 C4S7ET 57392007 IC50 > 100 nM T58992 CHSW27 57392492 IC50 = 0.78 nM T58992 CX89LJ 57392493 IC50 = 0.7 nM T58992 CJ38ZY 57393448 Ki > 10000 nM T58992 C9K0MG 57393724 IC50 = 23 nM T58992 C2V7SB 57393725 IC50 = 5.2 nM T58992 C6D7UA 57394195 IC50 = 0.2 nM T58992 C3K5FX 57394196 IC50 = 200 nM T58992 C4QZH8 57394197 IC50 = 0.2 nM T58992 CASY82 57394218 EC50 = 1.77 nM T58992 C2VWR5 57394219 EC50 = 0.19 nM T58992 CS02AB 57395174 Ki = 7200 nM T58992 CSE78X 57395267 IC50 = 0.67 nM T58992 C9CI3A 57395445 IC50 = 0.068 nM T58992 CZ9G4Q 57395446 IC50 = 0.78 nM T58992 C6SUR4 57395447 IC50 = 0.7 nM T58992 C4NI1O 57395962 IC50 = 0.16 nM T58992 C3BR0J 57396943 Ki > 15000 nM T58992 C12ASH 57396944 Ki > 7800 nM T58992 C9W6IB 57397288 IC50 = 0.9 nM T58992 CP0A2G 57397289 IC50 = 6.6 nM T58992 CG8O2H 57397290 IC50 = 1.1 nM T58992 CB7XV5 57397291 IC50 = 0.094 nM T58992 CNX73U 57397760 IC50 = 0.082 nM T58992 CC8EV2 57397761 IC50 = 0.75 nM T58992 C1HF3V 57397762 IC50 = 0.27 nM T58992 C84EKV 57398678 IC50 = 0.26 nM T58992 CSW1C3 57398976 IC50 = 1.4 nM T58992 C0JIL8 57398977 IC50 = 2 nM T58992 CP8KQ7 57399426 IC50 = 0.45 nM T58992 C4H6LZ 57399427 IC50 = 1.8 nM T58992 CLNB91 57399428 IC50 = 0.39 nM T58992 C7T9ID 57399429 IC50 = 0.17 nM T58992 C95NKZ 57400481 IC50 = 3.4 nM T58992 CMP1F7 57400482 IC50 = 0.63 nM T58992 CH13FG 57400694 IC50 = 0.29 nM T58992 C6W1SD 57400695 IC50 = 1.3 nM T58992 C3QF9I 57401062 Ki = 279 nM T58992 CU2V1C 57401137 IC50 = 4.7 nM T58992 CVXU49 57401184 IC50 = 0.22 nM T58992 C8RX7I 57402172 Ki = 5800 nM T58992 C5X0LN 57402288 IC50 = 0.46 nM T58992 CUL3W2 57402462 Ki > 1000 nM T58992 CJ0E6V 57402465 IC50 = 0.68 nM T58992 C6PM9O 57402466 IC50 = 0.26 nM T58992 CT1IN3 57412337 Ki = 290 nM T58992 C7F4PN 57412339 Ki = 730 nM T58992 CTO37U 57412341 Ki = 170 nM T58992 C0UZ3G 57412343 Ki = 530 nM T58992 CNI7Y9 57412772 Ki = 61 nM T58992 C21LRT 57412773 Ki = 150 nM T58992 CFB58K 57412848 Ki = 260 nM T58992 CTV4X5 57412849 Ki = 100 nM T58992 CSYI37 57412850 Ki = 53 nM T58992 CJI87G 57412851 Ki = 160 nM T58992 CCB0G9 57412852 Ki = 110 nM T58992 CDV4H9 57412853 Ki = 20 nM T58992 CAO20P 57412942 Ki = 150 nM T58992 CF1LC3 57412943 Ki = 110 nM T58992 CYN92K 57412944 Ki = 230 nM T58992 C54XQG 57412945 Ki = 120 nM T58992 C0GL5A 57412946 Ki = 30 nM T58992 CGN29J 57413036 Ki = 41 nM T58992 C5ZHT6 57413037 Ki = 13 nM T58992 CP9L1N 57413038 Ki = 720 nM T58992 CP6G5F 57413039 Ki = 190 nM T58992 CH0B1F 57413040 Ki = 350 nM T58992 CQW92S 57822038 Ki = 9.8 nM T58992 C8XF6W 57822045 Ki = 5.8 nM T58992 CV1Y9U 57822053 Ki = 11.8 nM T58992 CTE6B5 57822082 Ki = 6.8 nM T58992 CELJ49 57822098 Ki = 5.5 nM T58992 C60ZHX 57822157 Ki = 3.99 nM T58992 CK0P5N 57822243 Ki = 18 nM T58992 C0J3LY 57900041 Ki = 8.2 nM T58992 C6AWU4 57900045 Ki = 6.5 nM T58992 C67ZJA 57978865 EC50 = 103 nM T58992 C7MI3X 58046500 Ki > 10000 nM T58992 CFXC84 58046524 Ki > 10000 nM T58992 CI5H3N 58268566 Ki > 375 nM T58992 C6Z9JF 58268629 Ki > 400 nM T58992 C7EFU5 58443192 Ki = 1.9 nM T58992 C73BYR 58443217 Ki = 1.5 nM T58992 C5V8NC 58443218 Ki = 1.1 nM T58992 C7Z8SF 58443225 Ki = 0.81 nM T58992 CS70GT 58443229 Ki = 3.4 nM T58992 CFXB82 58443230 Ki = 3.9 nM T58992 C4FKN0 58443234 EC50 = 0.8 nM T58992 CW81HV 58443235 Ki = 0.55 nM T58992 CJO8H7 59345567 EC50 > 10000 nM T58992 C6GA5O 60150457 Ki > 10000 nM T58992 C7N0KO 60150458 Ki > 10000 nM T58992 C6G5TY 60154189 Ki > 400 nM T58992 C8MS6N 60154191 Ki > 400 nM T58992 CW63KM 60154192 Ki > 400 nM T58992 C2QX6R 60154193 Ki > 400 nM T58992 CD46EJ 60154264 Ki > 400 nM T58992 CEB0P5 60166738 Ki = 4751 nM T58992 CYUB94 60168107 Ki = 50010 nM T58992 CMAP25 60170608 Ki = 59290 nM T58992 C9AB5E 60170609 Ki = 56010 nM T58992 CQ3I4L 60170610 Ki = 10980 nM T58992 C9VYO5 60170611 Ki = 17040 nM T58992 CU35KA 60170688 Ki = 10810 nM T58992 CF8M6H 60170689 Ki = 5820 nM T58992 C2JUE9 60170691 Ki = 10200 nM T58992 C8U1DO 60170774 Ki = 18690 nM T58992 CW4P3F 60170775 Ki = 50930 nM T58992 CR1GS9 60170776 Ki = 84680 nM T58992 CY7E9U 60170777 Ki = 84850 nM T58992 CR50DU 67157108 Ki = 1.585 nM T58992 C87KCO 67182916 Ki = 12.59 nM T58992 C19UXP 67183276 Ki = 1.259 nM T58992 C1TEC7 67183439 Ki = 1.995 nM T58992 CF6RB3 67183527 Ki = 1.259 nM T58992 C5EV8P 67183538 Ki = 3.981 nM T58992 CNJ41I 67183562 Ki = 19.95 nM T58992 CY9R3L 67183680 Ki = 5.012 nM T58992 CYT8L5 67184545 Ki = 31.62 nM T58992 CM3JW0 67184580 Ki = 15.85 nM T58992 CYA6S5 67184933 Ki = 31.62 nM T58992 CZW53B 67933935 Ki = 113 nM T58992 C7KLB6 68196155 Ki = 2.5 nM T58992 C27KQI 68779363 Ki = 4300 nM T58992 C89TSB 68867300 Ki = 57.32 nM T58992 C4DO7H 70158365 Ki = 6 nM T58992 C30HMT 70681352 Ki > 10000 nM T58992 CS1E7F 70681353 Ki > 1000 nM T58992 C32MCZ 70682644 IC50 = 387 nM T58992 C5JLS9 70683421 Ki > 10000 nM T58992 CJ79UV 70683422 Ki > 10000 nM T58992 CH64DO 70683436 Ki > 10000 nM T58992 CZW6K5 70683437 Ki > 10000 nM T58992 CX3M0F 70683438 Ki > 5000 nM T58992 CXY52W 70685543 Ki > 10000 nM T58992 C60FVD 70685544 Ki > 10000 nM T58992 CU7V8F 70685545 Ki > 10000 nM T58992 CRKY09 70685720 IC50 = 262 nM T58992 CQL0S6 70687673 Ki > 10000 nM T58992 CY8DQ1 70687674 Ki > 10000 nM T58992 CE6K8V 70687698 Ki > 10000 nM T58992 CS86LY 70689742 Ki > 1000 nM T58992 CL3W2H 70691453 Ki = 4.4 nM T58992 CCQ5Z6 70691889 Ki > 1000 nM T58992 C1A7LO 70693567 Ki = 6.1 nM T58992 C9PQ4F 70693930 Ki > 10000 nM T58992 CMR2L1 70695247 IC50 = 111 nM T58992 CWO5F0 70695375 Ki > 400 nM T58992 CBM02Z 70696030 Ki = 1100 nM T58992 C2V8UI 70696034 Ki > 10000 nM T58992 CG3U7F 70697391 Ki > 400 nM T58992 CI8M5U 70834572 Ki > 10000 nM T58992 CEOQ43 71229805 Ki = 1.9 nM T58992 CIK86Q 71230334 Ki = 2.6 nM T58992 CLA6O8 71449105 IC50 > 8700 nM T58992 C2TY6U 71449133 Ki = 3.41 nM T58992 CEB0P4 71449173 IC50 = 13.2 nM T58992 C8HV9A 71449570 Ki > 5000 nM T58992 CQVN19 71449607 EC50 = 35 nM T58992 CYG07C 71449995 Ki = 75.3 nM T58992 CK69PO 71450043 Ki = 339.6 nM T58992 C4TVF1 71450063 Ki > 100000 nM T58992 CHQZ46 71450134 Ki = 2.71 nM T58992 CSC3R7 71450213 Ki = 2429 nM T58992 CJL59V 71450766 Ki = 2.2 nM T58992 C4BP5T 71450767 Ki = 0.9 nM T58992 C6JMZ4 71450851 Ki = 2.94 nM T58992 CQ6M2A 71450900 IC50 = 3442 nM T58992 C6ZX3S 71450925 Ki = 86.4 nM T58992 C5YIC1 71450926 Ki = 111 nM T58992 C2R7GS 71450927 Ki = 60.3 nM T58992 CMB7X9 71450932 Ki = 1.39 nM T58992 CNP02X 71450939 Ki = 4.6 nM T58992 C7FKC6 71451409 Ki = 1977 nM T58992 C3GX1O 71451410 Ki = 1230 nM T58992 C08KHB 71452040 Ki > 10000 nM T58992 C0XW8E 71452041 Ki > 10000 nM T58992 CO01JK 71452702 IC50 = 48 nM T58992 CYU3K7 71452742 Ki = 39 nM T58992 C4B6HU 71452746 EC50 = 0.33 nM T58992 CYFH30 71452786 IC50 = 3.8 nM T58992 C2YWE8 71453373 Ki = 14930 nM T58992 CQY10P 71453677 Ki = 103.9 nM T58992 CRY4A1 71453704 Ki > 100000 nM T58992 CYOS40 71453706 Ki > 100000 nM T58992 CW0H5Q 71453774 Ki = 17 nM T58992 CZ08WY 71454361 EC50 = 0.31 nM T58992 CG82PA 71454362 Ki = 1.5 nM T58992 CXD03J 71454425 IC50 = 20 nM T58992 CM0H5E 71454460 Ki > 10000 nM T58992 CGP4V5 71454476 IC50 = 13.9 nM T58992 CT60CU 71454481 IC50 = 11 nM T58992 CV4H8Q 71454482 IC50 = 5.5 nM T58992 CXQ1G0 71454513 Ki = 65.7 nM T58992 CGM86O 71454514 Ki = 5.38 nM T58992 CQ5JE8 71454515 Ki = 395 nM T58992 CI16ON 71454516 Ki = 741.55 nM T58992 CO01LV 71454517 Ki = 2.36 nM T58992 C09IMN 71454521 Ki > 10000 nM T58992 CYC5K3 71454539 Ki = 33 nM T58992 CCKA54 71454553 IC50 = 5.8 nM T58992 CYJ9X8 71454554 IC50 = 1080 nM T58992 CG96HQ 71454569 Ki = 27 nM T58992 CNL95W 71454964 EC50 = 20 nM T58992 CI0G3P 71455268 Ki > 10000 nM T58992 CN3EX8 71455429 Ki > 100000 nM T58992 CW63BC 71455505 Ki = 3.74 nM T58992 C89UMR 71455506 EC50 = 0.59 nM T58992 CFBC49 71455896 Ki = 5168 nM T58992 C83WJY 71456105 Ki = 6.6 nM T58992 CQ0UG3 71456106 EC50 = 0.16 nM T58992 CF9HA1 71456174 Ki = 27.8 nM T58992 CBM7U2 71456180 IC50 = 6.6 nM T58992 C7MIO2 71456181 IC50 = 1.4 nM T58992 C94HLU 71456182 IC50 = 36 nM T58992 C6QM8Z 71456225 IC50 = 25 nM T58992 C75DZW 71456227 IC50 = 2.9 nM T58992 C42HSQ 71456256 Ki = 10.3 nM T58992 C8FXZ5 71456257 EC50 = 0.87 nM T58992 CDQM86 71456258 Ki = 2.07 nM T58992 CXZ2V8 71456262 Ki = 0.08 nM T58992 C1G7OM 71456308 IC50 = 571 nM T58992 C2X3AN 71456309 IC50 > 10000 nM T58992 C42MER 71457207 Ki = 12.1 nM T58992 C3XIP8 71457209 Ki > 100000 nM T58992 C9UVJ1 71457210 Ki > 100000 nM T58992 CLN75C 71457288 Ki = 1.95 nM T58992 CH4Y5I 71457289 Ki = 1.63 nM T58992 CPUO14 71457290 Ki = 1.33 nM T58992 C4KD6E 71457291 Ki = 4.13 nM T58992 C0R8UO 71457292 Ki = 0.96 nM T58992 CDSX56 71457372 Ki = 3572 nM T58992 C53UEV 71457978 IC50 = 19 nM T58992 C9GQO5 71458037 IC50 > 10000 nM T58992 CSJ4A1 71458063 Ki = 6.53 nM T58992 CG98LJ 71458064 Ki = 4.83 nM T58992 CV74RO 71458065 EC50 = 1.4 nM T58992 C5SM7K 71458085 Ki = 746 nM T58992 CP6DQ7 71458116 IC50 = 12.1 nM T58992 C92YCB 71458142 IC50 = 122 nM T58992 CQ46CG 71458581 Ki = 1557 nM T58992 C8LNZ6 71459067 Ki > 100000 nM T58992 C7X9YH 71459820 Ki = 0.8 nM T58992 CA1N5D 71459821 Ki = 1.2 nM T58992 CU7EL6 71459888 IC50 = 1030 nM T58992 CNCA72 71459902 Ki = 10.97 nM T58992 CQ52LR 71459947 Ki = 94.1 nM T58992 CFR1T9 71459948 Ki = 289 nM T58992 CUID52 71459949 Ki = 87.9 nM T58992 C0TP7N 71459950 Ki = 322 nM T58992 CHS4D2 71459951 Ki = 8 nM T58992 CE2VA0 71459952 Ki = 38.6 nM T58992 CBHT09 71459962 Ki = 0.16 nM T58992 C6NOP7 71459993 EC50 = 28 nM T58992 C6IG5K 71460019 IC50 = 81.7 nM T58992 C12KHQ 71460850 Ki = 419.9 nM T58992 CJ65RV 71460942 Ki = 1.2 nM T58992 CC25XY 71460943 Ki = 1.78 nM T58992 CT52OM 71460944 EC50 = 0.27 nM T58992 C6NLR9 71460945 Ki = 0.97 nM T58992 CBEV63 71461579 Ki > 10000 nM T58992 CV60JN 71461663 Ki = 246 nM T58992 CFHE81 71461664 Ki = 133 nM T58992 CXT37B 71461665 Ki = 11.1 nM T58992 CY28RA 71461666 Ki = 7.59 nM T58992 C3O5EC 71461667 Ki = 2.88 nM T58992 C9Q6GY 71461668 EC50 = 7.53 nM T58992 CD4Q0A 71461673 Ki = 2.7 nM T58992 C9AJ6X 71461674 Ki = 0.27 nM T58992 C75JTH 71462114 Ki = 2254 nM T58992 C6N1FP 71462554 Ki = 160.4 nM T58992 C4ZD8G 71462655 Ki = 1.91 nM T58992 CB3L8W 71462656 Ki = 87 nM T58992 C2I5MZ 71463280 Ki = 0.84 nM T58992 CW8ZV5 71509717 EC50 = 0.43 nM T58992 CV72DZ 71509871 EC50 = 0.43 nM T58992 C8D1CB 71605418 Ki = 2810 nM T58992 CJ8GA4 71605419 Ki = 2780 nM T58992 CT3YS1 71605420 Ki = 5580 nM T58992 C4UG0T 71605421 Ki = 6950 nM T58992 C9Z7AT 71605588 Ki = 27.3 nM T58992 CG8ZD6 71605589 Ki = 19.8 nM T58992 CU53FL 71605755 Ki = 18.9 nM T58992 CMZ8F3 71605756 Ki = 30.4 nM T58992 CIW95L 71613507 Ki = 4320 nM T58992 C26ORE 71613508 Ki > 10000 nM T58992 CHI7D3 71613509 Ki > 10000 nM T58992 CEO5Z2 71613709 Ki > 10000 nM T58992 C8X6TP 71613710 Ki > 10000 nM T58992 C82MIG 71613711 Ki > 10000 nM T58992 C0MC1V 71613712 Ki > 10000 nM T58992 CVC5H1 71613903 Ki > 10000 nM T58992 CX9PM4 71613904 Ki > 10000 nM T58992 C2BOG7 71613905 Ki > 10000 nM T58992 CAJ61F 71613906 Ki > 10000 nM T58992 CS3CN1 71613907 Ki > 10000 nM T58992 C8XIJ1 71624166 Ki = 0.63 nM T58992 C2P7KV 71624167 Ki = 84 nM T58992 CSQ58W 71624287 Ki = 590 nM T58992 CH1X9Y 71624288 Ki = 0.28 nM T58992 C9D8EK 71624409 Ki = 24 nM T58992 CAT6R2 71624412 Ki = 36000 nM T58992 CRO68A 71624413 Ki = 13000 nM T58992 CH3M7S 71624446 Ki = 0.34 nM T58992 CJ2Z3X 71624447 Ki = 0.42 nM T58992 CASE43 71625485 Ki = 12 nM T58992 CBUK06 71625600 Ki = 630 nM T58992 C04BRZ 71625601 EC50 = 5.9 nM T58992 C38SBH 71625714 EC50 = 2.2 nM T58992 C8J7NS 71625715 Ki = 1000 nM T58992 CPS8A6 71625832 EC50 = 0.34 nM T58992 C2GF7U 71625833 Ki = 4.6 nM T58992 CDB6W2 71625948 Ki = 0.35 nM T58992 CBT73M 71625949 Ki = 0.51 nM T58992 C1A9BS 71660039 Ki = 64 nM T58992 CE0AX8 71660040 Ki = 36 nM T58992 CE5J8U 71660041 Ki = 29 nM T58992 CF4NS6 71660042 Ki = 75 nM T58992 CWBH85 71660081 Ki > 10000 nM T58992 CWKO96 71660082 Ki = 479 nM T58992 CXZ1D7 71660083 Ki = 207 nM T58992 CJK9R5 71660084 Ki = 33 nM T58992 C7R1TA 71660085 Ki = 128 nM T58992 C4U5ZF 71660086 Ki = 52 nM T58992 C64TPF 71660087 Ki = 39 nM T58992 CM6I2K 71660088 Ki = 111 nM T58992 CD9CN8 71660125 Ki = 34 nM T58992 CDS7T3 71660126 Ki = 26 nM T58992 C1AIY3 71660127 Ki = 26 nM T58992 CJ43VK 71660128 Ki = 24 nM T58992 CF57LR 71660129 Ki = 55 nM T58992 C58SAC 71660130 Ki = 136 nM T58992 CG7UJ9 71660163 Ki = 63 nM T58992 C5XM1H 71680922 Ki = 94.54 nM T58992 CUW3Z8 71680923 Ki = 39.88 nM T58992 CWSC46 71680924 Ki = 10.86 nM T58992 CP5FK9 71681076 Ki = 25.07 nM T58992 C4LV9A 71681077 Ki = 15.13 nM T58992 CE0YC8 71681078 Ki = 1.48 nM T58992 CU57ZQ 71681079 Ki = 10.54 nM T58992 CVM39A 71716193 IC50 > 30000 nM T58992 CG15IY 71717290 IC50 = 24 nM T58992 CM3PS4 71718530 IC50 = 32 nM T58992 CI0L2X 71719111 IC50 = 6.2 nM T58992 CZ8CL2 71719454 Ki = 22.2 nM T58992 CWZA14 71719730 IC50 = 198 nM T58992 C3LUG2 71720208 Ki = 0.49 nM T58992 CTU9Q8 71720326 IC50 = 5.3 nM T58992 CIZ7P6 71720342 IC50 = 7997 nM T58992 CY89EO 71720682 Ki = 25.6 nM T58992 CCB3X2 71726555 Ki = 2.1 nM T58992 C4G5IU 71726685 Ki = 3 nM T58992 CLBE62 71726686 Ki = 0.95 nM T58992 CU47GC 71751564 Ki = 5 nM T58992 CYR84C 71762505 Ki = 0.43 nM T58992 C0L7TE 71769137 Ki > 10000 nM T58992 CTX84S 71769138 Ki > 10000 nM T58992 C3YAR9 71769139 Ki > 10000 nM T58992 CWK9E7 71769267 Ki > 10000 nM T58992 C7G3EX 71769268 Ki > 10000 nM T58992 CEZW27 71769269 Ki = 6200 nM T58992 CMZ94S 71818133 EC50 = 0.26 nM T58992 CAMG13 71818134 Ki = 5.7 nM T58992 CZM8U6 71818277 Ki = 4.7 nM T58992 CW95UP 71819400 EC50 = 3200 nM T58992 C0EBP2 71819401 EC50 = 80 nM T58992 C7SQL1 71819402 EC50 = 13000 nM T58992 C8HK9Y 71819403 EC50 = 100000 nM T58992 C2MD4G 71819404 EC50 = 79000 nM T58992 CW0YD6 71819525 EC50 = 2500 nM T58992 CI4CE3 71819526 EC50 = 16000 nM T58992 C7W2PU 72163557 Ki = 695 nM T58992 CMZ9E5 72163689 Ki = 187 nM T58992 CVJC81 72163691 Ki = 1347 nM T58992 C4MA6E 72163693 Ki = 463 nM T58992 CZM45H 72163695 Ki = 1650 nM T58992 C05KYU 72163804 Ki = 2798 nM T58992 CS4RF2 72163806 Ki = 922 nM T58992 CQHB67 72202465 Ki = 551 nM T58992 CZQ86Y 72374835 Ki = 1961 nM T58992 CAK42B 72374836 Ki = 876 nM T58992 CWH6T3 72548703 IC50 = 6 nM T58992 C7NB1W 72711408 Ki = 0.65 nM T58992 C89COK 72711409 Ki = 4.6 nM T58992 C7FI6P 72711410 Ki = 1.6 nM T58992 C29YGC 72712370 EC50 = 750 nM T58992 CYEJ30 72713098 EC50 = 14.8 nM T58992 CJT7L9 72713099 Ki = 264 nM T58992 C4MWE1 72713100 Ki = 73.8 nM T58992 CPY8F1 72713101 Ki = 43.2 nM T58992 CBVG86 72713102 Ki = 18.4 nM T58992 CLRX12 72713104 Ki = 9.04 nM T58992 CC6Q5R 72771081 Ki < 100 nM T58992 CC65OA 73213195 Ki > 10000 nM T58992 CW83DK 73213196 Ki > 10000 nM T58992 COL97Y 73295685 IC50 = 3500 nM T58992 CNA8O3 73345364 Ki = 6030 nM T58992 CMU18J 73345366 Ki = 13500 nM T58992 CRAP90 73345445 Ki = 1020 nM T58992 CU6J4D 73345484 IC50 = 2340 nM T58992 CBD57O 73345518 Ki = 2.88 nM T58992 C1VW7Q 73345526 Ki = 7.4 nM T58992 C7ZN1K 73345634 Ki = 2041.74 nM T58992 CC4Z8N 73345675 IC50 = 850 nM T58992 CJV51U 73345676 IC50 = 2700 nM T58992 CIHT26 73345677 IC50 = 900 nM T58992 C53MQR 73345678 IC50 = 1400 nM T58992 C7VT4S 73345679 IC50 = 150 nM T58992 CCN72S 73345747 IC50 = 717 nM T58992 C6ML2U 73345882 Ki = 4600 nM T58992 C2KLJ6 73345883 Ki = 1.1 nM T58992 CY03SQ 73346599 Ki = 544 nM T58992 CU7C6J 73346891 Ki = 6760 nM T58992 CS01BP 73347048 Ki = 0.38 nM T58992 CS5F3B 73347271 Ki = 0.035 nM T58992 CQJ36Z 73347341 Ki > 10000 nM T58992 CH2T1I 73347643 Ki = 583 nM T58992 C5HXL6 73347644 Ki = 318 nM T58992 C0J9VP 73348396 IC50 = 2190 nM T58992 CMC60F 73348468 Ki = 57.7 nM T58992 CG12ZL 73348469 Ki = 24.8 nM T58992 C4YFP5 73348534 Ki = 1000 nM T58992 CEN4T7 73348535 Ki = 320 nM T58992 CD4YH3 73348548 Ki = 0.76 nM T58992 C97OCV 73348687 IC50 = 2400 nM T58992 C46QVZ 73348688 Ki > 10000 nM T58992 CENY03 73348689 IC50 = 285 nM T58992 CAE78D 73348734 Ki = 11 nM T58992 C37EDC 73348784 IC50 = 7.4 nM T58992 CUW07Z 73349067 Ki = 57 nM T58992 CA98UC 73349068 Ki = 250 nM T58992 CM70YA 73349151 Ki = 721 nM T58992 C9Z3KC 73349647 Ki = 438 nM T58992 C6S9GN 73350058 Ki = 42.4 nM T58992 CVEP75 73350098 IC50 = 1360 nM T58992 C0Z9UB 73350099 IC50 = 717 nM T58992 CBJ82D 73350102 IC50 = 245 nM T58992 C57VAX 73350104 IC50 = 2000 nM T58992 C80THJ 73350137 Ki = 27.8 nM T58992 C5IJO1 73350142 Ki = 7.8 nM T58992 CTE81Z 73350143 Ki = 11 nM T58992 CR9FM2 73350171 IC50 = 181 nM T58992 CWH52D 73350639 Ki = 9.3 nM T58992 C5GAW0 73351393 Ki = 5.2 nM T58992 CB42RH 73351424 Ki = 920 nM T58992 CMC83R 73351578 IC50 = 13 nM T58992 C63MRZ 73351589 IC50 = 242 nM T58992 CVM0A9 73351608 Ki = 84.3 nM T58992 CR2L8V 73351611 Ki = 2800 nM T58992 C0W1NT 73351837 IC50 = 2720 nM T58992 CQXJ82 73351885 EC50 = 239 nM T58992 CG27HN 73351999 EC50 = 0.22 nM T58992 CWA73N 73352217 Ki = 126 nM T58992 CL2W3H 73352233 Ki = 260 nM T58992 CSY9E4 73352234 EC50 = 3200 nM T58992 C7D1LF 73352661 Ki = 750 nM T58992 CL8HW5 73353046 IC50 = 18 nM T58992 C3HRP2 73353056 IC50 = 319 nM T58992 CAVE73 73353057 IC50 = 232 nM T58992 CRGW21 73353090 Ki = 0.66 nM T58992 C7OFK3 73353093 Ki = 1300 nM T58992 C3PZE0 73353313 IC50 = 4320 nM T58992 C9B6ZY 73353598 Ki = 0.2 nM T58992 C29SQL 73353599 Ki = 0.38 nM T58992 C2YO7N 73353600 Ki = 5.5 nM T58992 CKFA02 73353693 Ki = 139 nM T58992 C2NXP4 73354381 Ki = 370 nM T58992 C0JIR8 73354382 Ki = 35 nM T58992 CO3ZS7 73354458 Ki = 3230 nM T58992 C0SBM2 73354619 Ki = 21.6 nM T58992 C0P8YG 73354621 Ki = 113 nM T58992 CN1H6S 73354622 Ki = 28 nM T58992 CSL34I 73354623 Ki = 1.21 nM T58992 COS31U 73354624 Ki = 2340 nM T58992 C2SDM9 73354631 Ki = 110 nM T58992 CV6C8I 73354763 IC50 = 1980 nM T58992 C1BU3H 73354764 IC50 = 510 nM T58992 C6QAC3 73354765 IC50 = 300 nM T58992 CA8MQ1 73354785 Ki = 0.91 nM T58992 CA74SC 73354965 Ki = 4 nM T58992 CT34BM 73354966 Ki = 2.8 nM T58992 CORH63 73355099 Ki = 0.76 nM T58992 C2HJ6O 73355223 Ki = 116 nM T58992 C3Z5LT 73355419 Ki = 2787 nM T58992 CE6I8C 73355784 IC50 = 34 nM T58992 C3Q9FB 73356023 Ki = 15000 nM T58992 CM2U0C 73356135 IC50 = 53 nM T58992 C92ILU 73356142 IC50 = 15.9 nM T58992 C18PAF 73356143 IC50 = 1000 nM T58992 C1RZ8E 73356166 Ki = 430 nM T58992 CP87QL 73356293 IC50 = 440 nM T58992 CM57TY 73356294 IC50 = 2120 nM T58992 C5PB4R 73356663 Ki = 130 nM T58992 C83ZPI 73356767 Ki = 103 nM T58992 CJT8Y2 73356768 Ki = 3540 nM T58992 C2LZD4 76309826 Ki = 0.37 nM T58992 CB78KL 76309827 Ki = 117.4 nM T58992 C68BLJ 76309828 Ki = 170.3 nM T58992 C35USC 76313542 EC50 = 3.2 nM T58992 C6J2WF 76313543 Ki = 10.9 nM T58992 CZSU65 76313544 Ki = 15.1 nM T58992 C1GU9H 76317053 Ki = 818.4 nM T58992 CM9RC0 76317054 Ki = 57.3 nM T58992 CSYN97 76317055 Ki = 1.48 nM T58992 C0SWX7 76317056 Ki = 9.1 nM T58992 CP95SN 76317057 Ki = 22.8 nM T58992 CPKY85 76320762 Ki = 405.3 nM T58992 CG9MB3 76324401 Ki = 0.43 nM T58992 CU12ZJ 76324412 Ki = 160.5 nM T58992 CIX43W 76327982 Ki > 10000 nM T58992 CB4JI7 76331634 Ki = 907.2 nM T58992 CCW07O 76331635 EC50 = 19.7 nM T58992 CRA1Y0 76331636 Ki = 10.5 nM T58992 C6F1BS 76335253 EC50 = 14.2 nM T58992 COK40D 76335254 Ki = 3.92 nM T58992 CZP08R 76335255 Ki > 10000 nM T58992 CM27VY 78210001 Ki = 208 nM T58992 CTI5S8 81689720 Ki = 0.941 nM T58992 C97GYK 89435126 EC50 = 0.35 nM T58992 CL5R0T 89435196 Ki = 0.356 nM T58992 C7X1VI 89435275 Ki = 1.26 nM T58992 C08YSC 89435280 Ki = 0.833 nM T58992 CZSC16 90306849 EC50 = 0.64 nM T58992 C03HOW 90392373 Ki = 0.154 nM T58992 C0OAE4 90392376 EC50 = 0.42 nM T58992 C47BLH 90397724 Ki = 0.211 nM T58992 C54EUB 90644257 Ki = 1.1 nM T58992 CZ10JE 90644258 Ki = 31.6 nM T58992 CV7U4P 90644259 Ki = 1.88 nM T58992 CI2TV6 90644873 Ki = 8 nM T58992 C3WD0A 90644874 Ki = 2.1 nM T58992 CGBL95 90644875 Ki = 0.49 nM T58992 C9B0JT 90645382 IC50 > 1000 nM T58992 C3VIY8 90645383 IC50 > 1000 nM T58992 C6YPT9 90645384 IC50 > 1000 nM T58992 CPB25R 90645385 IC50 > 1000 nM T58992 C18HBT 90645386 IC50 > 1000 nM T58992 C1DOG7 90654745 Ki > 375 nM T58992 CX3WT1 90654746 Ki > 375 nM T58992 CC70MH 90654747 Ki > 375 nM T58992 C4ZQD5 90654748 Ki > 375 nM T58992 CBV23K 90654749 Ki > 375 nM T58992 C87NYV 90654750 Ki > 375 nM T58992 C20FOK 90654751 Ki > 375 nM T58992 CT91LC 90654752 Ki > 375 nM T58992 C1Y6QN 90655511 IC50 < 100 nM T58992 CIQV28 90655825 EC50 = 15.6 nM T58992 C6V1PS 90655826 EC50 = 2 nM T58992 CNPC03 90655827 EC50 = 9.2 nM T58992 CFAZ39 90655828 EC50 = 0.39 nM T58992 C63YPH 90655829 EC50 = 0.41 nM T58992 C6FN2S 90656087 Ki = 475 nM T58992 C2QY3H 90656088 Ki = 221 nM T58992 CW2P5Q 90656089 Ki = 1060 nM T58992 C8TV7C 90656090 EC50 > 5000 nM T58992 CK9FP8 90656664 Ki = 1.2 nM T58992 CC6LY3 90656665 EC50 = 1.76 nM T58992 COGW86 90656666 Ki = 0.86 nM T58992 C9YKV8 90656667 Ki = 1.2 nM T58992 C3WLH8 90656668 Ki = 0.8 nM T58992 C4A3CZ 90663908 Ki = 24 nM T58992 CW91YF 90663910 Ki = 5.7 nM T58992 CP1ZW6 90663949 Ki > 5000 nM T58992 CZ9GL5 90663950 Ki > 5000 nM T58992 CFK27M 90663951 Ki > 5000 nM T58992 CBT6F1 90663952 Ki > 5000 nM T58992 C1QAB3 90663953 Ki = 222 nM T58992 C3QA8Z 90664881 EC50 = 7.5 nM T58992 C5VZC6 90666479 Ki = 108 nM T58992 C2NG3A 90666726 Ki > 10000 nM T58992 C5DG9V 90666727 Ki > 10000 nM T58992 C26HUP 90666728 Ki > 10000 nM T58992 CK0W6U 90666729 Ki > 10000 nM T58992 CM75TG 90666730 Ki > 5000 nM T58992 C4D6WT 90666731 Ki > 5000 nM T58992 C0GWK7 90666732 Ki > 5000 nM T58992 CT70RV 90666733 Ki > 5000 nM T58992 CT0O1B 90666734 Ki > 10000 nM T58992 CCUK67 90666735 Ki > 10000 nM T58992 CWI2S7 90666736 Ki > 3000 nM T58992 C0BNE6 90667279 Ki = 2 nM T58992 CWOB91 90667280 Ki = 2 nM T58992 CU2XP8 91801212 EC50 = 52.7 nM T58992 CR93LZ 91928491 Ki = 860 nM T58992 C2UZ4P 91928492 Ki = 1010 nM T58992 C07VRA 101341769 Ki > 10000 nM T58992 CI4YM3 101806592 EC50 = 83.7 nM T58992 CYUT97 101880775 Ki = 12 nM T58992 CW3LH2 101882818 Ki = 37.2 nM T58992 CW5H9D 101882819 Ki = 2486 nM T58992 CGQV37 101882820 Ki = 2607 nM T58992 CNHS29 101898709 IC50 = 1690 nM T58992 CO5Z0L 102014213 Ki = 24.8 nM T58992 CPT9B3 102269996 Ki = 1.58 nM T58992 C9T1NI 102269998 Ki = 0.85 nM T58992 COFT20 102270003 Ki = 0.92 nM T58992 CR4KN5 102270004 Ki = 2.85 nM T58992 CP5F4Q 102270005 Ki = 9.25 nM T58992 C3FX4P 102270006 Ki = 1.02 nM T58992 CFA7K6 102270007 Ki = 3.59 nM T58992 CD19TA 102270008 Ki = 9.39 nM T58992 C8P4XF 117705986 EC50 = 3 nM T58992 C0BCI6 117705988 EC50 = 0.61 nM T58992 CEP48V 117706009 Ki = 0.221 nM T58992 CMO27R 117706010 Ki = 0.501 nM T58992 C67SPE 117706054 Ki = 0.265 nM T58992 C12FIV 117706085 Ki = 1.46 nM T58992 CSJ3H4 117860306 EC50 = 1.4 nM T58992 C3A7QZ 118200491 Ki = 115.9 nM T58992 CR52EZ 118200640 Ki = 179.2 nM T58992 CUCJ65 118263805 IC50 = 4410 nM T58992 C9JV1T 118263857 IC50 > 10000 nM T58992 CRY49P 118263892 IC50 > 10000 nM T58992 C9YVS2 118263923 IC50 > 10000 nM T58992 C5HCS3 118264001 IC50 > 10000 nM T58992 C38LHY 118264112 IC50 = 2410 nM T58992 CM8TB4 118705898 Ki = 0.36 nM T58992 C6RW0E 118705901 Ki = 0.28 nM T58992 C8ZM3D 118709349 Ki > 100000 nM T58992 C58BHC 118709350 Ki > 100000 nM T58992 C01ZSF 118709356 Ki > 100000 nM T58992 CK3S0G 118709357 Ki > 100000 nM T58992 CIJX58 118709358 Ki > 100000 nM T58992 CN3UC7 118709360 Ki > 100000 nM T58992 CI1QT3 118711134 IC50 = 3380 nM T58992 C4MRB0 118711135 IC50 > 100000 nM T58992 CP6WQ1 118711209 IC50 > 100000 nM T58992 CL9F4B 118711887 Ki = 169 nM T58992 CBK60I 118713122 Ki > 10000 nM T58992 C5J0UN 118713123 Ki = 2625 nM T58992 CJ38GQ 118713124 Ki > 10000 nM T58992 CCIS67 118713125 Ki > 10000 nM T58992 CDU9H7 118713126 Ki = 3260 nM T58992 C8TPM0 118713127 Ki > 10000 nM T58992 C9E8OS 118713128 Ki = 3032 nM T58992 CRVW31 118713129 Ki = 700.5 nM T58992 CO8UJ6 118713130 Ki > 10000 nM T58992 CL25HD 118713131 Ki > 10000 nM T58992 CI52KQ 118713132 Ki > 10000 nM T58992 C5MJX6 118713133 Ki > 10000 nM T58992 C4MHO8 118713134 Ki > 10000 nM T58992 CT7EU4 118713135 Ki > 10000 nM T58992 CZFQ32 118713136 Ki > 10000 nM T58992 C0P3QL 118713137 Ki > 10000 nM T58992 CE4Z7B 118713138 Ki > 10000 nM T58992 C14HFW 118713139 Ki > 10000 nM T58992 C7HO5D 118713140 Ki = 5871 nM T58992 C7NHP9 118713141 Ki = 4888 nM T58992 CUY58S 118713142 Ki = 228.2 nM T58992 C78LKO 118716009 EC50 = 1.7 nM T58992 C5BJA6 118716010 EC50 > 1000 nM T58992 C30HPC 118718754 Ki = 100 nM T58992 CKQ94A 118718755 Ki = 26 nM T58992 CEG97T 118718757 Ki = 50 nM T58992 C34ULN 118718758 Ki = 110 nM T58992 CET8O5 118718759 Ki = 200 nM T58992 C5XTV8 118718760 Ki = 86 nM T58992 C0OT5D 118718761 Ki = 27 nM T58992 C8SUW9 118718762 Ki = 6.4 nM T58992 C2BCI6 118718763 Ki = 7.8 nM T58992 C69JPI 118718764 Ki = 700 nM T58992 C0SY6C 118718765 Ki = 42 nM T58992 C29GAH 118719100 Ki = 16.3 nM T58992 CU10SI 118722557 EC50 = 42.5 nM T58992 CA51CQ 118724536 Ki > 5000 nM T58992 CH4LB0 118724977 Ki > 5000 nM T58992 C9SN0M 118724979 Ki > 5000 nM T58992 CH9GT5 118724980 Ki > 5000 nM T58992 CG7SQ8 118724984 Ki > 5000 nM T58992 C29CVM 118725741 EC50 = 1800 nM T58992 C0HM6Y 118725745 EC50 = 5500 nM T58992 CXL16I 118725841 EC50 = 1700 nM T58992 C49YCX 118725843 EC50 = 100000 nM T58992 CCQ85P 118725848 EC50 = 5200 nM T58992 C1Q5IB 118725849 EC50 = 100000 nM T58992 CE86DJ 118725850 EC50 = 2800 nM T58992 CBDA90 118725853 EC50 = 12 nM T58992 CET5Y3 118725854 EC50 = 72 nM T58992 C2LA6F 118725855 EC50 = 82 nM T58992 CO8B9L 118725856 EC50 = 1850 nM T58992 CMO86W 118725857 EC50 = 37000 nM T58992 C61VHK 118725858 EC50 = 1150 nM T58992 CFNX71 118726846 Ki = 72.81 nM T58992 C5LUM4 118726847 Ki = 254.16 nM T58992 C5MSK4 118726848 Ki = 81.33 nM T58992 CT0O1J 118726849 Ki = 72.92 nM T58992 CQH1G3 118731120 Ki = 4.2 nM T58992 CDN86Z 118731405 Ki = 6.9 nM T58992 CK5W7M 118731406 Ki = 15 nM T58992 C29ESD 118731407 Ki = 13 nM T58992 CAP48T 118731408 Ki = 7.1 nM T58992 C12NJU 118731409 Ki = 18 nM T58992 CM06BI 118731410 Ki = 9.1 nM T58992 CP84KM 118731411 Ki = 5.5 nM T58992 C5MK1D 118731412 Ki = 229 nM T58992 CPD5R9 118731413 Ki = 116 nM T58992 CY9NH0 118731414 Ki = 7.3 nM T58992 CR6K5D 118731415 Ki = 21 nM T58992 CMR93J 118731416 Ki = 26 nM T58992 CQ39OA 118731417 Ki = 57 nM T58992 CK76UL 118731418 Ki = 21 nM T58992 CRXY76 118731419 Ki = 16 nM T58992 C9A4RX 118731420 Ki = 589 nM T58992 CC2S7I 118731421 Ki = 68 nM T58992 C3N0VC 118731422 Ki = 148 nM T58992 C4FT8K 118731423 Ki = 25 nM T58992 C1L4QH 118731424 Ki = 44 nM T58992 CB0R9K 118731425 Ki = 54 nM T58992 CW35DR 118731426 Ki = 127 nM T58992 CP61XB 118731427 Ki = 24 nM T58992 CD51ZQ 118731428 Ki = 719 nM T58992 CIP6E1 118731878 EC50 = 23 nM T58992 CNT5W9 118737392 EC50 = 1000 nM T58992 CUT4V5 118737393 EC50 = 100 nM T58992 CT24GR 118737394 EC50 = 50 nM T58992 C19VKC 118737395 EC50 = 200 nM T58992 CSL4C7 118737396 EC50 = 300 nM T58992 C59YKQ 118737397 EC50 = 900 nM T58992 C5SAR8 118737398 EC50 = 1000 nM T58992 CR1L6M 118737399 EC50 > 10000 nM T58992 CWO42N 121365644 Ki > 10000 nM T58992 CG52CR 121365655 Ki = 5190 nM T58992 C9ND2K 121373679 Ki = 2328 nM T58992 C0J9GQ 121432154 Ki = 6.31 nM T58992 C6KIU4 121614638 IC50 = 40 nM T58992 CWP9E2 122178420 EC50 = 125.89 nM T58992 CQ7YP3 122178421 EC50 = 162.18 nM T58992 C31KTI 122178424 EC50 = 9.333 nM T58992 C5JCY2 122178425 EC50 = 33.88 nM T58992 C1A2JB 122178426 EC50 = 8.71 nM T58992 CRKB15 122179557 EC50 = 457.09 nM T58992 C93YZC 122179560 EC50 = 51.29 nM T58992 C70SUR 122181051 EC50 = 6365 nM T58992 CN0S6Q 122181052 EC50 = 1639 nM T58992 CO04MC 122181110 EC50 = 366 nM T58992 C3UV6A 122182776 Ki = 2.71 nM T58992 CVMP98 122182777 Ki = 1.11 nM T58992 C20HCF 122182778 Ki = 1.94 nM T58992 C3S5RY 122182780 Ki = 15.5 nM T58992 C18PTI 122182782 EC50 = 45.5 nM T58992 C6R8UI 122182784 EC50 = 6.71 nM T58992 CG7N6Q 122182786 Ki = 2.77 nM T58992 CYJ34R 122182788 Ki = 5.58 nM T58992 CDJ0N9 122182790 Ki = 18.2 nM T58992 CWYQ85 122182792 Ki = 37.8 nM T58992 C80PUY 122183206 Ki = 1400 nM T58992 CP7G1A 122183208 Ki = 840 nM T58992 C6GLF5 122183209 Ki = 1200 nM T58992 CIP5Y3 122183210 Ki = 2300 nM T58992 C9YU5A 122183211 Ki = 1500 nM T58992 CMR9Q4 122183213 Ki = 430 nM T58992 C0CPO2 122183218 Ki = 9.2 nM T58992 CDUW32 122183219 Ki = 3.6 nM T58992 CA7R3L 122183220 Ki = 31 nM T58992 C7EO2T 122183221 Ki = 21 nM T58992 C7QKU8 122183222 Ki = 73 nM T58992 CA0B9X 122183223 Ki = 6.6 nM T58992 CXE52Q 122183281 Ki = 15 nM T58992 CV0FU5 122183282 Ki = 4.2 nM T58992 CEP3K5 122183283 Ki = 17 nM T58992 CB9Z1T 122183284 Ki = 3.8 nM T58992 CVH6E0 122187205 EC50 = 0.38 nM T58992 CP20LG 122187206 EC50 = 3.4 nM T58992 C7JS5O 122187722 Ki = 11 nM T58992 C27RVE 122187723 EC50 = 6.7 nM T58992 CTO0D6 122187724 Ki = 0.8 nM T58992 CJ8D0B 122187725 EC50 = 24 nM T58992 C6FV7P 122189395 Ki = 6000 nM T58992 COJT48 122189396 IC50 = 0.2754 nM T58992 C0Y9GD 122189397 Ki > 10000 nM T58992 CV5RT0 122189398 Ki = 7800 nM T58992 C2YB4V 122189399 Ki = 5700 nM T58992 C6TW5C 122189401 Ki > 10000 nM T58992 CTM75I 122189402 Ki = 10000 nM T58992 C9ERU6 122189403 Ki > 10000 nM T58992 CDVT64 122189404 Ki > 10000 nM T58992 CVSA53 122189405 Ki > 10000 nM T58992 CI8ND7 122189406 Ki > 10000 nM T58992 C0NEX5 122189407 Ki = 5200 nM T58992 CM1UE8 122189409 Ki = 4500 nM T58992 C0F9BP 122189854 Ki > 10000 nM T58992 C6HN2A 122189855 Ki = 6900 nM T58992 C8EP5B 122189856 Ki > 10000 nM T58992 CG7Q1O 122189857 Ki = 1700 nM T58992 CHUO37 122189858 Ki = 36 nM T58992 C4QJ3S 122189859 Ki = 2 nM T58992 CD04RY 122189860 Ki = 38 nM T58992 CBD35W 122189861 Ki = 7 nM T58992 CUAF39 122189862 Ki = 2 nM T58992 CRWT03 122189863 Ki = 3 nM T58992 CCO3N2 122189901 Ki = 0.2 nM T58992 C4OUQ0 122190289 Ki = 320 nM T58992 CM2L5X 122190290 Ki = 720 nM T58992 C60CBH 122190291 Ki = 370 nM T58992 CW64DN 122190292 Ki = 34 nM T58992 CO56JT 122190293 Ki = 0.5 nM T58992 CS64OW 122194218 Ki = 12050 nM T58992 CS1IN2 122194219 Ki = 13280 nM T58992 CNE13U 122194668 Ki = 3.72 nM T58992 CCQ3E0 122197314 IC50 > 5700 nM T58992 C5K8XH 122197315 IC50 > 10000 nM T58992 CFWE98 122197316 IC50 > 10000 nM T58992 CZ03XS 122197485 IC50 = 3800 nM T58992 C0WTE6 122197486 IC50 = 5300 nM T58992 C1TP0H 122197487 IC50 = 2900 nM T58992 CSN3V4 122197488 IC50 > 10000 nM T58992 C6LC2J 122197489 IC50 > 8800 nM T58992 CPCF21 122197490 IC50 = 3300 nM T58992 CF8X5R 122197491 IC50 > 4700 nM T58992 CMA83V 122197492 IC50 = 460 nM T58992 CX4I7N 122197493 IC50 = 1300 nM T58992 CWZA97 122197494 IC50 > 10000 nM T58992 CTKY87 122197495 IC50 > 10000 nM T58992 CH9O2Q 122197496 IC50 = 8840 nM T58992 C5I8CM 122197497 IC50 > 7800 nM T58992 C7EF4P 122197498 IC50 = 2040 nM T58992 C1BDZ4 122197499 IC50 = 49 nM T58992 C7F8CK 122197500 IC50 > 10000 nM T58992 CMH7K2 122197501 IC50 > 10000 nM T58992 CD3L6S 122197502 IC50 > 10000 nM T58992 C7O1EP 122197503 IC50 = 7500 nM T58992 CYE18M 122197504 IC50 = 2500 nM T58992 C9W2FQ 122197505 IC50 = 530 nM T58992 C45VUL 122197506 IC50 = 4040 nM T58992 CEP3J0 122197507 IC50 = 5020 nM T58992 C9B5DC 122197508 IC50 > 10000 nM T58992 CZTO90 122197509 IC50 > 9700 nM T58992 C7SJO2 122197510 IC50 > 10000 nM T58992 CH93LB 122197511 IC50 = 6630 nM T58992 CL78AV 122197512 IC50 = 890 nM T58992 CAQ5B0 122409965 Ki = 3100 nM T58992 C0K8BS 122589938 Ki = 2178 nM T58992 CBU38O 122589952 Ki = 2129 nM T58992 CTNU73 123445395 Ki = 29 nM T58992 C8OXG3 127024961 Ki = 0.259 nM T58992 CZ5NJ7 127025173 Ki = 4.79 nM T58992 C9FBD2 127025219 Ki = 0.48 nM T58992 CL3VG1 127025528 Ki = 1 nM T58992 CRDW90 127026456 EC50 = 64.57 nM T58992 CO5S0Z 127026457 EC50 = 53.7 nM T58992 C6D7EV 127028324 Ki = 0.44 nM T58992 CW6RV7 127028653 Ki = 0.16 nM T58992 CO7H8W 127029282 Ki = 0.94 nM T58992 CIW9F7 127029283 Ki = 0.75 nM T58992 C8AO1V 127029284 Ki = 0.021 nM T58992 CSK04O 127032208 Ki = 0.531 nM T58992 CR3TB5 127032209 Ki = 0.303 nM T58992 C2SP1T 127032210 Ki = 2.3 nM T58992 CXJY65 127032211 Ki = 2.76 nM T58992 CK29CG 127032212 Ki = 0.644 nM T58992 CQ25BG 127032213 Ki = 0.585 nM T58992 CN0BZ9 127033398 Ki = 12.1 nM T58992 CFR46S 127033399 Ki = 0.0945 nM T58992 CML91J 127033967 EC50 = 1.83 nM T58992 CZ61LK 127034966 EC50 > 5011.87 nM T58992 CA0SN5 127034967 EC50 > 5011.87 nM T58992 CT8C3S 127034976 EC50 = 6600 nM T58992 C4WGV3 127034992 Ki = 0.6 nM T58992 C4MN9G 127035664 Ki = 2 nM T58992 C1PQ2T 127035665 Ki = 0.2 nM T58992 C31BZD 127035666 Ki = 1.2 nM T58992 CEV3A7 127036745 Ki = 5200 nM T58992 C6F8CK 127036746 Ki = 9000 nM T58992 C0LO8V 127037378 Ki = 5200 nM T58992 CFBS45 127037395 Ki = 8950 nM T58992 C8HYD4 127037396 Ki = 5900 nM T58992 C5ODE6 127037397 Ki = 3702 nM T58992 CX6P8G 127037398 Ki = 3700 nM T58992 CKL40H 127037399 Ki = 4100 nM T58992 CCE7L8 127037400 Ki = 5800 nM T58992 CWIQ78 127037438 Ki = 0.4 nM T58992 CXMJ48 127043001 Ki = 194 nM T58992 CSV07U 127043062 Ki > 10000 nM T58992 C0CMH9 127043073 Ki > 10000 nM T58992 C3W5SX 127043074 Ki > 10000 nM T58992 CQVP14 127043075 Ki > 10000 nM T58992 C32KON 127043249 Ki > 10000 nM T58992 C7CKP3 127043256 Ki > 10000 nM T58992 C7XF0S 127043262 Ki > 10000 nM T58992 C5GU8A 127043275 Ki = 4.7 nM T58992 CFU4H9 127043364 Ki = 85 nM T58992 CUX47D 127043424 Ki > 10000 nM T58992 CCP2Z8 127043425 Ki = 140 nM T58992 C7HM0D 127043432 Ki = 720 nM T58992 C0WM8J 127043433 Ki = 160 nM T58992 C8CV6X 127043434 Ki = 65 nM T58992 C30BNK 127043559 Ki = 117 nM T58992 C1GK3A 127043614 Ki = 260 nM T58992 C61FHR 127043615 EC50 = 2.6 nM T58992 CCSZ68 127044528 Ki = 99 nM T58992 C4CW7A 127047717 Ki = 5800 nM T58992 C4SU9L 129093829 Ki > 1000 nM T58992 C1EHU5 129188443 Ki = 923 nM T58992 CD8FT9 129188454 Ki = 1690 nM T58992 CC9Z0J 129188459 Ki = 3070 nM T58992 CWQO32 132584396 Ki > 10000 nM T58992 CENF10 132584397 Ki > 10000 nM T58992 CM1PN3 132584398 Ki > 10000 nM T58992 CS2H6B 132584403 Ki > 10000 nM T58992 CAVB41 132584404 Ki > 10000 nM T58992 CSK3I8 132609309 EC50 = 58.88 nM T58992 C0NUC2 132609310 EC50 = 14.45 nM T58992 C9Z6XL 132609311 EC50 = 95.5 nM T58992 CO69MW 134130798 Ki > 10000 nM T58992 CA1V9U 134131635 Ki > 10000 nM T58992 C4GPT2 134131885 Ki > 10000 nM T58992 C3Z6SV 134131949 Ki > 10000 nM T58992 C64JNH 134134355 Ki > 10000 nM T58992 C91TWF 134134844 Ki > 10000 nM T58992 C7A1PO 134137537 Ki > 10000 nM T58992 CL4K1Z 134139120 Ki > 10000 nM T58992 CK2X3O 134139232 Ki > 10000 nM T58992 C80ZPT 134139387 Ki > 10000 nM T58992 CSX32C 134141708 Ki > 10000 nM T58992 CC8V6M 134142063 Ki > 10000 nM T58992 CTQ91W 134142390 Ki > 10000 nM T58992 CG0V4O 134142896 Ki > 10000 nM T58992 CBG64F 134144504 Ki > 10000 nM T58992 CU3L0J 134145684 Ki > 10000 nM T58992 CGV52O 134147031 Ki = 2187 nM T58992 C5VAD3 134147144 Ki > 10000 nM T58992 C62SOQ 134147564 Ki > 10000 nM T58992 C8DP6W 134147710 Ki > 10000 nM T58992 CB8CI0 134147910 Ki > 10000 nM T58992 CBU81N 134149168 Ki > 10000 nM T58992 C5ZD9L 134149737 Ki > 10000 nM T58992 CH97MA 134154487 Ki > 10000 nM T58992 CT2X3N 134155538 Ki > 10000 nM T58992 C9QBY4 134156534 Ki > 10000 nM T58992 C13PHC 134157413 Ki > 10000 nM T58992 CLS5H3 134227139 Ki = 18.9 nM T58992 CG57MT 134563466 Ki = 4067 nM T58992 CE5RS7 134563496 Ki > 10000 nM T58992 CAEY19 134563500 Ki > 10000 nM T58992 C82SEF 134563650 Ki > 10000 nM T58992 CC3HK6 134563655 Ki > 10000 nM T58992 C4U9EM 134563691 Ki > 10000 nM T58992 CFX37T 134563695 Ki = 2712 nM T58992 CPEH72 134563698 Ki > 10000 nM T58992 CR74XA 134563699 Ki > 10000 nM T58992 C9PN6I 134578342 Ki > 10000 nM T58992 CK62WY 134578456 Ki > 10000 nM T58992 CN0C9Z 134578457 Ki > 10000 nM T58992 C0HNI9 134578506 Ki = 6028 nM T58992 C0JCQ2 134578518 Ki > 10000 nM T58992 CGN13V 134611895 Ki = 941 nM T58992 C1GY2T 135156251 EC50 > 10000 nM T58992 CPZ89B 135314564 Ki > 1000 nM T58992 CAX4E7 135329044 IC50 > 10000 nM T58992 CG7P3W 135329090 IC50 > 10000 nM T58992 CMS56H 135329094 IC50 > 10000 nM T58992 CUYV98 135329104 IC50 > 10000 nM T58992 CRW47P 135329122 IC50 > 10000 nM T58992 CWE6O8 136126655 Ki = 780 nM T58992 C8IP5C 136126656 Ki = 2000 nM T58992 CQKN40 137434120 IC50 > 10000 nM T58992 C0PL4B 137434175 IC50 = 6500 nM T58992 CNCS34 137434196 IC50 > 10000 nM T58992 CW8LH6 137434204 IC50 > 10000 nM T58992 COQ5H7 137434366 IC50 > 10000 nM T58992 C2JK8N 137434496 IC50 = 4500 nM T58992 CVBP38 137541794 IC50 = 4180 nM T58992 C3QB8I 137541808 IC50 = 170 nM T58992 CW6SK2 137541816 IC50 = 190 nM T58992 C0BKU3 137631438 Ki > 10000 nM T58992 CTH8M9 137631847 Ki = 1432 nM T58992 CFT36I 137631943 Ki = 1.585 nM T58992 CB0IT4 137632188 Ki = 158.49 nM T58992 C9WUL6 137632260 Ki > 1000 nM T58992 CNC15K 137632903 Ki > 10000 nM T58992 C6FEL8 137633728 Ki = 8.64 nM T58992 C4SR3G 137633741 Ki = 316.23 nM T58992 CX37GF 137633920 Ki = 6.31 nM T58992 C7D9QE 137634365 Ki = 3.981 nM T58992 CBW57P 137634403 Ki = 1862 nM T58992 COJ2S3 137634747 Ki = 3.162 nM T58992 CB14RN 137635022 Ki = 83.9 nM T58992 C8QAR1 137636327 Ki = 1.259 nM T58992 C5EO6T 137637552 Ki = 429.3 nM T58992 CN07MB 137637586 Ki = 1.995 nM T58992 C5CTQ7 137638063 Ki = 1.259 nM T58992 COS82Q 137638460 Ki = 3.981 nM T58992 C3NT7A 137638511 Ki = 4.19 nM T58992 CKR9S7 137638688 Ki = 2268 nM T58992 C4CWP3 137639680 Ki = 266.6 nM T58992 CBM34G 137640362 Ki = 1.585 nM T58992 CUZ7O1 137640860 Ki = 1469 nM T58992 CY2AV8 137641064 Ki = 168 nM T58992 C2OD0K 137641318 Ki > 1000 nM T58992 CMI3T0 137641479 IC50 = 15.82 nM T58992 CF7Q8M 137641618 Ki = 12.9 nM T58992 C1RAK0 137642012 Ki = 2775 nM T58992 CID94R 137642522 Ki = 25.12 nM T58992 C1IAZ5 137642772 Ki = 18.1 nM T58992 CKH93R 137643506 Ki > 10000 nM T58992 CAI9Z4 137643649 Ki > 10000 nM T58992 CU7MG5 137644005 Ki = 100 nM T58992 C2MRK0 137645329 Ki > 1000 nM T58992 CX7UD0 137645396 Ki = 0.5012 nM T58992 CG4N0O 137646080 Ki = 14.4 nM T58992 C2OB5H 137646522 Ki > 10000 nM T58992 CXJ9G7 137646782 Ki = 1637 nM T58992 CY1R8I 137646935 Ki = 79.43 nM T58992 C3MV2Q 137646937 Ki = 489.4 nM T58992 CTP82Z 137647554 Ki = 3539 nM T58992 CQ76TD 137648147 Ki = 2.512 nM T58992 CX72UG 137648224 Ki = 76.7 nM T58992 CK8EP7 137648628 Ki = 85.5 nM T58992 CH8F7A 137649449 Ki = 49.6 nM T58992 C4TDX9 137649850 Ki = 2743 nM T58992 CBC86L 137650237 Ki = 0.5012 nM T58992 CZ68WR 137651510 Ki = 738 nM T58992 CV4Y7Q 137652968 Ki = 0.7943 nM T58992 CK74TN 137652971 Ki = 2.15 nM T58992 C9YHQ5 137653349 Ki = 67 nM T58992 CS1B3U 137654001 Ki = 1312 nM T58992 C6N8JM 137655206 Ki = 428 nM T58992 C7P9UA 137655599 Ki = 2139 nM T58992 C3KPA4 137655663 Ki = 84 nM T58992 CSHN48 137656887 Ki = 2850 nM T58992 CY21WB 137657032 EC50 = 0.23 nM T58992 CWD31I 137657725 Ki = 0.89 nM T58992 CG8R9U 137660781 Ki > 10000 nM T58992 CR0EW1 137660824 Ki = 3340 nM T58992 C1XPN8 137661045 Ki > 1000 nM T58992 CNX2Q5 137662177 Ki > 1000 nM T58992 C9LM6E 137662178 Ki = 1099 nM T58992 CH6X3W 140995821 Ki = 3162.28 nM T58992 CZ82RG 145948744 Ki = 5 nM T58992 C3EWL2 145948797 Ki = 1 nM T58992 CMD58S 145948809 Ki = 13 nM T58992 C2RLY9 145948839 Ki = 4 nM T58992 CGA46O 145948847 Ki = 1 nM T58992 CHGW16 145948955 Ki = 260 nM T58992 C7N5LP 145948965 Ki = 14 nM T58992 CH49XK 145948968 Ki = 7 nM T58992 CCB85T 145948980 Ki = 160 nM T58992 C5E2QA 145948981 Ki = 5 nM T58992 C16WUV 145949356 Ki = 250 nM T58992 CDA24L 145950961 Ki > 100000 nM T58992 CE9SQ4 145952136 IC50 = 58 nM T58992 CM17OA 145952209 IC50 = 100 nM T58992 C7WT1M 145952813 Ki > 100000 nM T58992 C4V7GC 145952964 IC50 = 68 nM T58992 CVZ04C 145956193 Ki = 1130 nM T58992 C9Y8RW 145956549 IC50 = 94 nM T58992 C7SX5C 145957352 Ki > 100000 nM T58992 C7X0LW 145958562 Ki > 100000 nM T58992 CI9XG5 145958618 IC50 = 76 nM T58992 CW2T8U 145959553 IC50 = 58 nM T58992 CY1MB9 145961131 Ki = 1.9 nM T58992 CR8WC1 145961165 Ki = 3.981 nM T58992 CIU2V6 145961844 Ki = 0.46 nM T58992 CGR0Y1 145963106 Ki = 25.12 nM T58992 CBFE94 145963594 Ki = 1.995 nM T58992 CH0VD5 145964426 Ki > 10000 nM T58992 C2MS3R 145966170 Ki = 1470 nM T58992 CB2WA9 145972038 Ki = 3260 nM T58992 CQS9N0 145978012 Ki = 940 nM T58992 C87MSW 145980271 Ki = 10000 nM T58992 C63FHK 145982510 Ki = 123.2 nM T58992 C36TEU 145982515 Ki = 160.3 nM T58992 CC6A9H 145982585 Ki = 1490 nM T58992 CU2IK5 145982792 Ki = 55.4 nM T58992 CTQV67 145982828 Ki = 349.4 nM T58992 C8MY6V 145982968 Ki = 485.4 nM T58992 CO8Z4U 145983526 Ki = 26.3 nM T58992 C4L7PT 145983969 Ki = 59.3 nM T58992 CK6F1J 145984022 Ki = 48.6 nM T58992 C1ONP2 145984192 Ki = 263.9 nM T58992 COP2I9 145984332 Ki = 773.7 nM T58992 C4KS7H 145984702 Ki = 345 nM T58992 CTY73C 145984984 Ki = 103.6 nM T58992 C4N3JP 145986165 Ki = 127.1 nM T58992 CNJH37 145986752 Ki = 10000 nM T58992 CUGO10 145988693 Ki = 1558 nM T58992 C0FT8Y 145991902 Ki = 3.31 nM T58992 C2ADQ5 145994326 EC50 = 0.53 nM T58992 C3CP1R 145994327 EC50 = 1.055 nM T58992 CFO47R 145994330 EC50 = 6.02 nM T58992 CBFX85 145994331 EC50 = 3.32 nM T58992 CF7GX6 145994332 EC50 = 1.932 nM T58992 CL69BD 145994333 EC50 = 1.952 nM T58992 CSE72Q 145994334 EC50 = 0.7787 nM T58992 CW6I7K 145994336 EC50 = 1.217 nM T58992 C0YWU3 145994337 EC50 = 1.408 nM T58992 CVK19A 145994338 EC50 = 1.637 nM T58992 CT3MY4 145994339 EC50 = 1.085 nM T58992 C23IEG 145994341 EC50 = 2.305 nM T58992 CZC6W1 145994342 EC50 = 2.522 nM T58992 C9RJO2 145994343 EC50 = 1.351 nM T58992 CG9XC0 145994345 EC50 = 6.644 nM T58992 C6P3SR 153287553 Ki > 10000 nM T58992 CV9G7Z 153287572 Ki > 10000 nM T58992 CO85KL 153287574 Ki > 10000 nM T58992 CL6OY2 155510745 Ki = 7.3 nM T58992 CVMK78 155512747 Ki = 50 nM T58992 CG95UQ 155512955 Ki = 106 nM T58992 CEV36D 155513829 Ki = 16.83 nM T58992 CKRG27 155513884 Ki = 29 nM T58992 C6F2GE 155514186 Ki = 1.2 nM T58992 C1UXA4 155514661 Ki = 2.4 nM T58992 CKL4N0 155515090 IC50 > 10000 nM T58992 CTHA56 155515703 Ki = 29.79 nM T58992 CSM5N3 155515838 Ki = 2900 nM T58992 CUM2N4 155515982 Ki = 10000 nM T58992 C0U6OJ 155516255 EC50 = 43 nM T58992 C7RT4P 155516535 Ki = 5.9 nM T58992 C3MQP5 155516545 Ki = 74 nM T58992 C3PD8O 155516811 Ki = 2.7 nM T58992 CJ80FA 155516945 IC50 > 10000 nM T58992 C2Z4UD 155517287 EC50 = 587 nM T58992 C7TD1C 155517330 Ki = 2.04 nM T58992 C5HXW8 155518735 Ki > 100000 nM T58992 C27NLG 155518912 Ki = 35.9 nM T58992 CUSA24 155519891 Ki > 10000 nM T58992 CF42WX 155520785 EC50 = 1995.26 nM T58992 CY5CL2 155521553 Ki > 10000 nM T58992 C7QCK2 155522403 EC50 = 5 nM T58992 CZ9V8E 155522689 Ki = 1400 nM T58992 CWA8B7 155523094 Ki = 4.8 nM T58992 CUYJ91 155524409 Ki = 18.65 nM T58992 C24PLM 155525923 Ki > 1000 nM T58992 C4O3FT 155526173 Ki = 12.26 nM T58992 C9L5FR 155526451 Ki = 1.39 nM T58992 C69DEY 155526658 Ki = 30.67 nM T58992 CDFR34 155526934 EC50 = 1.4 nM T58992 C1SZ3R 155527414 IC50 > 10000 nM T58992 C5B7LS 155527564 Ki = 31 nM T58992 C7T5YS 155527675 Ki = 3.162 nM T58992 CMZK90 155528037 Ki = 5.31 nM T58992 CV42PH 155529675 Ki = 39 nM T58992 CE36BU 155530150 Ki = 6.85 nM T58992 C1FW6M 155530357 Ki = 7900 nM T58992 CXH95L 155531153 Ki > 10000 nM T58992 CUD59P 155531529 Ki = 10.29 nM T58992 CJS61X 155531666 Ki = 38.93 nM T58992 C6W5JY 155532087 Ki = 5257 nM T58992 C3UV2R 155532761 Ki = 1.585 nM T58992 CV0UL2 155532879 Ki = 1 nM T58992 C7GU3F 155533321 Ki = 12.59 nM T58992 CEG3N8 155533730 Ki > 100000 nM T58992 C5S8MZ 155535351 Ki = 1.259 nM T58992 CB79ZW 155536080 Ki > 10000 nM T58992 C2YV1C 155536562 EC50 = 4.3 nM T58992 CE6Q7N 155536593 IC50 = 0.36 nM T58992 CZT05I 155537442 Ki = 7.943 nM T58992 CR97JX 155537513 Ki = 10620 nM T58992 CSZK58 155538263 Ki = 25.12 nM T58992 C61NAO 155538316 Ki = 16.91 nM T58992 CYEL64 155539136 Ki = 43 nM T58992 CE8UF7 155539181 Ki = 3.08 nM T58992 CPDK87 155539216 Ki = 280 nM T58992 C5NE1H 155539282 Ki = 900 nM T58992 CX86BV 155539726 Ki = 15.7 nM T58992 CI26FJ 155540400 EC50 > 10 nM T58992 CJF25T 155540464 Ki = 2.1 nM T58992 C0ML6F 155542107 Ki = 19.95 nM T58992 CJV8E5 155542270 Ki = 2.512 nM T58992 C67WLH 155542684 Ki > 10000 nM T58992 CA27KR 155543816 IC50 > 10000 nM T58992 C27SCO 155543969 Ki = 1.995 nM T58992 C57JHT 155544775 Ki = 70.55 nM T58992 CK36RG 155545176 Ki = 12666 nM T58992 CGKR14 155546429 EC50 = 5 nM T58992 CGJ1T5 155546569 Ki = 157 nM T58992 C6HGY8 155547045 Ki = 31 nM T58992 CKAN65 155549973 IC50 > 10000 nM T58992 CDFU45 155549997 EC50 = 8.1 nM T58992 C5H7AI 155551063 Ki = 19.95 nM T58992 C4S7MG 155551744 IC50 > 10000 nM T58992 CX8JA1 155552185 Ki = 19000 nM T58992 C0WH2Y 155552342 Ki > 100000 nM T58992 CHSX69 155552921 Ki = 10 nM T58992 CLKV39 155554074 EC50 = 32.36 nM T58992 C81USE 155554575 Ki = 76 nM T58992 CHQ2X8 155554943 Ki = 9.9 nM T58992 CE2PJ9 155555050 EC50 = 4 nM T58992 CO1HJ8 155555908 Ki = 14.31 nM T58992 C2BX9P 155556076 Ki = 22.28 nM T58992 C2TD1R 155558095 IC50 = 2000 nM T58992 CPW10R 155558236 Ki = 11.87 nM T58992 CH3E0B 155558313 Ki = 47 nM T58992 CODF60 155558752 Ki = 2900 nM T58992 C8GSZ2 155559127 Ki = 1.36 nM T58992 CF3U0D 155559400 IC50 = 900 nM T58992 C61BFO 155559678 Ki = 44.4 nM T58992 CKI47R 155560346 Ki = 63.1 nM T58992 C20UAD 155561395 Ki > 100000 nM T58992 CQ6G9E 155563096 Ki = 34 nM T58992 CJT89K 155563204 IC50 > 10000 nM T58992 CAN0G3 155563660 Ki > 1000 nM T58992 C9QN6H 155563763 Ki = 9.07 nM T58992 C3A6ZY 155563934 Ki = 440 nM T58992 C4AXT9 155564059 Ki = 18.9 nM T58992 COL80P 155564087 Ki = 24.04 nM T58992 C6C7IM 155564346 Ki = 1.94 nM T58992 CWG3K0 155565050 Ki = 5.012 nM T58992 CIS95O 155565113 Ki = 193 nM T58992 CEZ16B 155565184 Ki > 100000 nM T58992 CUQ25H 155566579 Ki = 4.94 nM T58992 CL76VI 155566581 Ki = 1.93 nM T58992 C2H6EK 155567280 Ki = 17.56 nM T58992 CZ89CL 155567972 Ki = 8.35 nM T58992 C2MV4D 155568748 Ki = 199.53 nM T58992 CTNU54 155569410 Ki = 0.82 nM T58992 CQ0GL3 155569552 Ki > 10000 nM T58992 C3N9VU 10251906 Ki > 500 nM T58992 CP9TR0 10324985 Ki > 10000 nM T58992 CVDX02 13935836 Ki = 28.84 nM T58992 C9FSE0 14015071 Ki = 18.04 nM T58992 CLF5U2 15005472 Ki = 43.6 nM T58992 C0X2QM 15005475 Ki = 158 nM T58992 C0VBY2 18666969 Ki > 10000 nM T58992 CFR6A5 46905974 Ki = 170 nM T58992 CAB94M 5484063 Ki = 18 nM T58992 D00FXL 44439907 Ki = 3.8 nM T58992 D00JPB 44434951 Ki = 2.86 nM T58992 D00NRB 6602241 Ki = 0.62 nM T58992 D00NZP 44447368 EC50 > 1000 nM T58992 D00SDP 44627900 Ki = 5.4 nM T58992 D00TNR 5311081 EC50 > 1000 nM T58992 D00XZH 44430025 Ki = 52825 nM T58992 D00YCW 44426807 Ki = 4126 nM T58992 D01ADK 11693641 Ki = 85 nM T58992 D01AQC 9811733 Ki = 1 nM T58992 D01EPU 9804450 Ki = 1.3 nM T58992 D01GYS 44377415 IC50 = 0.475 nM T58992 D01HOP 44439875 Ki = 170 nM T58992 D01MHO 44414725 Ki = 1152 nM T58992 D01MUV 10314141 Ki = 56600 nM T58992 D01RFG 10086063 Ki = 5.2 nM T58992 D01SDX 44439910 Ki = 1 nM T58992 D01TKS 10371120 Ki = 0.66 nM T58992 D01WMU 9820782 Ki = 5791 nM T58992 D02EIB 25129433 Ki = 59 nM T58992 D02IMZ 44427184 Ki = 15 nM T58992 D02NSY 10296561 IC50 > 10000 nM T58992 D02PIG 11250396 Ki = 1.8 nM T58992 D02RYZ 16083055 Ki = 1.5 nM T58992 D02YXR 10454860 Ki = 842 nM T58992 D03EPA 11051303 Ki = 0.2 nM T58992 D03KAQ 44626544 Ki > 10000 nM T58992 D03PTV 10022129 Ki = 898 nM T58992 D03RBD 49765077 IC50 = 8306 nM T58992 D03SAV 3082718 Ki = 24 nM T58992 D03UFD 5491897 Ki = 0.7 nM T58992 D03UHT 44429061 Ki = 360 nM T58992 D03UJW 22970051 Ki = 18800 nM T58992 D03VEQ 44377416 IC50 = 18.2 nM T58992 D03WGS 44408525 Ki = 23 nM T58992 D04EQE 46888571 IC50 = 2500 nM T58992 D04FBZ 5284595 Ki = 120 nM T58992 D04JCJ 44434931 Ki > 5000 nM T58992 D04JCK 644209 IC50 = 1.3 nM T58992 D04JFL 16099582 IC50 = 32 nM T58992 D04PPP 44406697 Ki = 9.4 nM T58992 D04QUB 25242485 Ki > 10000 nM T58992 D04RPI 16105563 EC50 = 29.3 nM T58992 D04SFK 644210 Ki = 0.48 nM T58992 D04UIK 44427178 Ki = 1.6 nM T58992 D04VJE 44434061 Ki = 2274 nM T58992 D04ZQX 44426812 Ki = 550 nM T58992 D05ANN 5486827 Ki = 0.013 nM T58992 D05COL 11440685 Ki > 10000 nM T58992 D05CRC 9909743 IC50 = 5.51 nM T58992 D05EWZ 44444966 Ki = 1.4 nM T58992 D05EXX 15764659 IC50 = 17000 nM T58992 D05EZE 10077295 Ki = 283 nM T58992 D05FEQ 5359966 Ki = 0.22 nM T58992 D05HOH 44447367 EC50 > 1000 nM T58992 D05JSY 10462426 Ki = 9.4 nM T58992 D05KIS 16100411 Ki = 0.8 nM T58992 D05MXI 42611190 Ki = 2750 nM T58992 D05QJS 5480230 Ki = 0.3 nM T58992 D05RII 44413409 Ki > 5000 nM T58992 D05XCV 44583427 Ki > 1000 nM T58992 D05ZIH 45110000 Ki = 213 nM T58992 D06BRA 11520765 EC50 = 128.82 nM T58992 D06DDA 46888587 IC50 = 5100 nM T58992 D06EES 461776 EC50 = 0.08 nM T58992 D06IXE 11411315 Ki = 730 nM T58992 D06KFX 44583372 Ki = 2000 nM T58992 D06MQG 44430018 Ki = 9585 nM T58992 D06NIP 11629355 Ki = 1500 nM T58992 D06NST 19143 Ki = 2 nM T58992 D06OKE 44427174 Ki = 53 nM T58992 D06PHT 10269001 Ki = 1666 nM T58992 D06PVO 44426806 Ki = 20890 nM T58992 D06QGJ 52946209 IC50 > 30000 nM T58992 D06XDA 16086543 IC50 = 1550 nM T58992 D06YMS 6917707 Ki = 1.3 nM T58992 D06YVE 44414877 Ki = 600 nM T58992 D07BPA 11645313 Ki = 1500 nM T58992 D07CIU 9924923 Ki = 12115 nM T58992 D07DFD 44427176 Ki = 42 nM T58992 D07FCB 9925737 Ki = 33110 nM T58992 D07GQE 10033203 Ki = 1.3 nM T58992 D07HFU 44429064 Ki = 50 nM T58992 D07ICW 11556976 Ki = 1.5 nM T58992 D07JIQ 44439882 Ki = 19 nM T58992 D07KTF 24873526 Ki = 1017 nM T58992 D07LQQ 11564210 Ki = 2.6 nM T58992 D07NMH 10093682 Ki = 15240 nM T58992 D07PPK 44406272 Ki = 81 nM T58992 D07QUY 44583388 Ki > 1000 nM T58992 D07UJV 44414785 Ki = 325 nM T58992 D08DVV 44430026 Ki = 17865 nM T58992 D08IWF 44427180 Ki = 30 nM T58992 D08IXN 5497186 Ki = 0.03 nM T58992 D08KSJ 24768351 EC50 = 35 nM T58992 D08LIT 11641503 Ki = 160 nM T58992 D08NJB 16733487 EC50 = 0.88 nM T58992 D08QBS 44178080 IC50 > 10000 nM T58992 D08QBU 44430029 Ki = 13750 nM T58992 D08QKT 11528076 Ki = 2 nM T58992 D08RPH 11255361 Ki = 180 nM T58992 D08SCK 11664525 Ki = 11 nM T58992 D08TFY 10043439 Ki = 8105 nM T58992 D08UZJ 12368881 Ki > 500 nM T58992 D09BWX 44583373 Ki > 1000 nM T58992 D09BYD 20481138 Ki = 1668 nM T58992 D09DUE 44429063 Ki = 160 nM T58992 D09EMR 11136782 EC50 = 128.82 nM T58992 D09FJY 9863568 Ki = 969 nM T58992 D09FLC 44627904 Ki = 160 nM T58992 D09GQP 15384271 IC50 = 1.6 nM T58992 D09GSD 11721803 Ki = 427 nM T58992 D09LRO 44430008 Ki = 5610 nM T58992 D09RJT 16086540 IC50 = 14600 nM T58992 D09RPR 16737207 Ki > 10000 nM T58992 D09RUY 44627790 Ki = 29 nM T58992 D09SBU 44583393 Ki > 1000 nM T58992 D09UKS 11303119 Ki = 230 nM T58992 D09VRT 44426814 Ki = 187 nM T58992 D0A3YH 24853671 EC50 = 960 nM T58992 D0A9AJ 44439901 Ki = 42 nM T58992 D0AC0A 10047612 Ki > 400 nM T58992 D0B8MY 9897164 Ki = 4.2 nM T58992 D0C1AN 44348645 IC50 = 230 nM T58992 D0C2UQ 44427183 Ki = 3.9 nM T58992 D0C6RQ 24768356 EC50 = 31 nM T58992 D0C7MP 44429062 Ki = 23 nM T58992 D0CK8C 24768352 EC50 = 31 nM T58992 D0D0UP 10315818 Ki = 8446 nM T58992 D0D0XP 44414814 Ki = 414 nM T58992 D0D1VB 11498201 EC50 > 1000 nM T58992 D0D3UB 45270599 EC50 = 0.06 nM T58992 D0D4AU 21593990 IC50 = 5500 nM T58992 D0D5QV 9838803 Ki = 2900 nM T58992 D0D5VD 44583375 Ki > 1000 nM T58992 D0D6OA 44414783 Ki = 18.8 nM T58992 D0D8AN 13374610 Ki = 79 nM T58992 D0D9BB 10427620 Ki = 45590 nM T58992 D0E0TD 44434950 Ki = 0.92 nM T58992 D0E2OG 11614928 Ki = 310 nM T58992 D0E6GH 44565511 Ki = 0.48 nM T58992 D0E6IT 44439879 Ki = 475 nM T58992 D0ED2I 11016572 Ki = 0.042 nM T58992 D0EM9A 107847 IC50 = 1.3 nM T58992 D0F1EB 44417373 Ki = 4.5 nM T58992 D0F1XY 44408590 Ki = 45 nM T58992 D0F4AN 44427182 Ki = 27 nM T58992 D0F8AX 44430024 Ki = 130550 nM T58992 D0F8CV 5462471 Ki = 0.66 nM T58992 D0FF6S 16038374 IC50 > 10000 nM T58992 D0FT5V 44583898 IC50 = 9900 nM T58992 D0G4FA 10384734 Ki = 19220 nM T58992 D0G4NM 104787 EC50 = 0.12 nM T58992 D0G6GC 25129135 Ki = 0.44 nM T58992 D0G7DF 44426827 Ki = 2437 nM T58992 D0G7FB 9798655 Ki = 29 nM T58992 D0H0KP 44434946 Ki = 495.99 nM T58992 D0H1BU 10864183 Ki = 0.031 nM T58992 D0H2CI 44456192 Ki = 2840 nM T58992 D0H3GI 25129090 Ki = 72 nM T58992 D0H3QK 44416393 IC50 = 13000 nM T58992 D0H6AA 44414843 Ki = 40 nM T58992 D0HB6O 44439880 Ki = 1 nM T58992 D0HN2M 44430609 Ki = 426.58 nM T58992 D0HQ0E 55652 Ki = 9400 nM T58992 D0I1BJ 16105560 EC50 = 3.55 nM T58992 D0I1NG 44434058 Ki = 0.97 nM T58992 D0I1ZN 44583428 Ki > 1000 nM T58992 D0I2CE 44583376 Ki = 670 nM T58992 D0I3XV 9840689 Ki = 0.355 nM T58992 D0I9PH 16100409 Ki = 2.2 nM T58992 D0IC5F 44414801 Ki = 1598 nM T58992 D0IL9H 44430013 Ki = 33345 nM T58992 D0IY2V 44429065 Ki = 270 nM T58992 D0J3NK 44427177 Ki = 2.8 nM T58992 D0J5JO 44430009 Ki = 7796 nM T58992 D0J7GJ 44408484 Ki = 1.4 nM T58992 D0J7VL 44439873 Ki = 1100 nM T58992 D0JH5D 44430007 Ki = 5610 nM T58992 D0K1BV 44628003 Ki = 320 nM T58992 D0K4XQ 44427175 Ki = 78 nM T58992 D0KW4Y 10485385 IC50 > 10 nM T58992 D0L2CT 24768355 EC50 = 72 nM T58992 D0L5DN 11392313 Ki = 150 nM T58992 D0L5MW 181743 Ki > 10000 nM T58992 D0L8LX 123704 Ki = 10 nM T58992 D0L8YY 10066285 Ki = 1720 nM T58992 D0L9YP 44254503 Ki = 17 nM T58992 D0M1YV 16747727 IC50 = 2740 nM T58992 D0M8YB 159059 IC50 = 11400 nM T58992 D0M9GO 115208 Ki = 153 nM T58992 D0N0JC 10808145 Ki = 1.07 nM T58992 D0N2DN 25129089 Ki = 71 nM T58992 D0N6DN 44408524 EC50 = 26.92 nM T58992 D0N6ZO 46888570 IC50 = 11300 nM T58992 D0NA7G 16083058 Ki = 4.2 nM T58992 D0NE3U 5485199 IC50 = 210 nM T58992 D0O1JD 44434057 Ki = 23.14 nM T58992 D0O6SB 443408 Ki = 0.23 nM T58992 D0O7JV 44426810 Ki = 184 nM T58992 D0OH7D 5310988 Ki = 2.81 nM T58992 D0P0RB 24768354 EC50 = 77 nM T58992 D0P2TT 73354725 Ki = 19 nM T58992 D0P3FP 44426808 Ki = 441 nM T58992 D0P5IH 44583387 Ki > 1000 nM T58992 D0P5QI 44626540 Ki = 1400 nM T58992 D0P6FF 44627901 Ki = 130 nM T58992 D0P8TI 11466688 Ki > 10000 nM T58992 D0PN3P 44439877 Ki = 10 nM T58992 D0Q1PN 44408417 EC50 = 0.5248 nM T58992 D0Q3XK 46888588 IC50 = 700 nM T58992 D0Q5AJ 44365804 Ki = 2500 nM T58992 D0Q6CF 44583374 Ki > 1000 nM T58992 D0Q7HG 24768353 EC50 = 10 nM T58992 D0Q9TQ 10043898 Ki = 2651 nM T58992 D0QH4A 10089987 Ki = 3325 nM T58992 D0QP2S 44408526 Ki = 0.82 nM T58992 D0R2VL 44434060 Ki > 5000 nM T58992 D0R4GI 11040230 Ki = 2.2 nM T58992 D0R4QF 11431898 Ki = 1170 nM T58992 D0R5TA 5311080 EC50 = 932 nM T58992 D0R6VF 6540640 IC50 = 0.19 nM T58992 D0R7LY 16733485 EC50 = 0.83 nM T58992 D0R9AP 44439872 Ki = 19 nM T58992 D0S2OA 10388166 Ki = 3741 nM T58992 D0S3TZ 5748293 Ki = 61.1 nM T58992 D0S5FN 44439876 Ki = 0.78 nM T58992 D0S7SO 16100407 Ki = 0.63 nM T58992 D0SC3W 44406704 Ki = 190 nM T58992 D0SE9S 9887077 Ki = 2854 nM T58992 D0T4ZY 44426817 Ki = 15250 nM T58992 D0T6OQ 10021946 Ki = 110 nM T58992 D0T9KE 44430016 Ki = 4392 nM T58992 D0TH8E 44414864 Ki = 15.2 nM T58992 D0TO0E 44467662 EC50 = 0.047 nM T58992 D0TR0U 10942040 Ki = 0.42 nM T58992 D0TT5V 44414811 Ki > 10000 nM T58992 D0U3ZL 23635044 Ki = 9400 nM T58992 D0U5OP 11580459 Ki = 140 nM T58992 D0U5QL 16040172 IC50 = 1650 nM T58992 D0U6OA 10909103 Ki = 0.22 nM T58992 D0U7JS 44439866 Ki = 1.3 nM T58992 D0U7PT 25075996 Ki = 3.8 nM T58992 D0UA3E 46888612 IC50 = 2100 nM T58992 D0UG5M 9956146 Ki = 29.6 nM T58992 D0UG8H 23642304 EC50 = 0.018 nM T58992 D0V0RB 11722088 EC50 = 4.074 nM T58992 D0V3OY 105104 Ki > 1000 nM T58992 D0V9DY 16100410 Ki = 1.1 nM T58992 D0VO7C 10677974 Ki = 2.9 nM T58992 D0W0CO 44627903 Ki = 39 nM T58992 D0W1YD 44439896 Ki = 360 nM T58992 D0W2DN 44427179 Ki = 2.7 nM T58992 D0W3VT 10091033 Ki = 6364 nM T58992 D0WT7H 5311018 Ki = 22.4 nM T58992 D0WZ7J 44414842 Ki = 154 nM T58992 D0X1SN 10010455 IC50 = 369 nM T58992 D0X2HT 44414863 Ki = 584 nM T58992 D0X4SX 10317947 Ki = 2767 nM T58992 D0X5TB 44439905 Ki = 1.2 nM T58992 D0X7LC 11061906 EC50 = 75.86 nM T58992 D0XX1Y 44426828 Ki = 9365 nM T58992 D0Y2HI 11635818 Ki = 27.2 nM T58992 D0Y5LJ 10336926 Ki = 14455 nM T58992 D0Y5ZP 44626534 Ki = 300 nM T58992 D0Y7CI 123924 Ki = 1.2 nM T58992 D0Y7KE 44430012 Ki = 24900 nM T58992 D0Y8NO 22977851 Ki = 12.6 nM T58992 D0YK5E 49860169 Ki = 69 nM T58992 D0YU5H 44434949 Ki = 27.6 nM T58992 D0Z6DK 44423026 IC50 = 13600 nM T58992 D0Z8JX 44583386 Ki = 3400 nM T58992 D0ZE2W 44430028 Ki = 15010 nM T99932 D09QEI 4740 IC50 = 85000 nM T99932 D0C4YC 4075 IC50 = 20600000 nM T99932 D05VZE 119031 IC50 = 1001 nM T99932 D0T5PO 5092 IC50 = 200 nM T99932 D07FHZ 5087 IC50 = 50000 nM T99932 D0T3ME 156422 EC50 = 18 nM T99932 CY9A0M 66065 IC50 = 12500 nM T99932 C21OTL 151419 IC50 > 200000 nM T99932 CQDJ34 428211 IC50 > 100000 nM T99932 CPE2J7 461663 IC50 = 12000 nM T99932 CNH7C2 461664 IC50 = 2900 nM T99932 C13KWU 461665 IC50 = 260000 nM T99932 C8PR3E 461666 IC50 = 380 nM T99932 CS3J5K 467265 IC50 = 400 nM T99932 C9YR0M 676987 IC50 = 200000 nM T99932 CZ37KX 874861 IC50 > 100000 nM T99932 CW9TZ3 1137620 IC50 > 100000 nM T99932 CDQ2E4 1367407 IC50 = 42300 nM T99932 C6O7AP 1582566 IC50 = 14000 nM T99932 C5CW1K 3081830 IC50 > 200000 nM T99932 CE80AQ 5327044 IC50 = 22000 nM T99932 CI13SQ 6523638 IC50 = 5750 nM T99932 C32HOB 9797095 IC50 = 150000 nM T99932 C2EV5L 9824551 IC50 = 10000 nM T99932 CJQ20V 9840218 IC50 = 120000 nM T99932 CF5T8E 9840925 IC50 = 7500 nM T99932 CF7AS4 9841064 IC50 = 51000 nM T99932 CX35SG 9850770 EC50 = 50 nM T99932 C34KGT 9892658 EC50 = 9 nM T99932 C13TVP 9904193 IC50 = 6000 nM T99932 CF1OJ6 9907022 IC50 = 70000 nM T99932 C49ILA 9936768 EC50 = 19 nM T99932 C2KI0C 9948975 IC50 = 3000 nM T99932 CFDN06 9949152 IC50 = 62000 nM T99932 C6XV8K 10019033 IC50 = 5000 nM T99932 C1NSK8 10091288 IC50 = 5600 nM T99932 CK5CJ9 10165915 EC50 = 42 nM T99932 CCE2T5 10229750 EC50 = 20 nM T99932 CBCW38 10256389 EC50 = 9 nM T99932 CV1WZ5 10301047 EC50 = 36 nM T99932 C1QM5I 10360825 IC50 = 60000 nM T99932 C4FOR3 10423517 IC50 = 4000 nM T99932 CL7N3F 10452587 IC50 = 450 nM T99932 CK3CH6 10498658 IC50 = 37000 nM T99932 C1BNW9 10498936 IC50 > 25000 nM T99932 CMTG10 10500152 IC50 > 100000 nM T99932 C1X5GM 10503011 IC50 = 11000 nM T99932 C49VUL 10515426 IC50 = 5000 nM T99932 CYH81M 10515726 IC50 > 200000 nM T99932 C3WQD5 10520713 IC50 = 15000 nM T99932 CZ8Y2I 10522445 IC50 = 38000 nM T99932 CY1V5H 10522585 IC50 = 15000 nM T99932 C63OLU 10527621 IC50 > 50000 nM T99932 C3S8WZ 10538504 IC50 = 55000 nM T99932 CI3GV1 10539258 IC50 > 25000 nM T99932 CN97DW 10539960 IC50 > 200000 nM T99932 C1HP3M 10541869 IC50 > 25000 nM T99932 CAKR74 10543322 IC50 = 35000 nM T99932 C2E0DT 10546983 IC50 = 175000 nM T99932 CB4QK3 10547110 IC50 = 1000 nM T99932 C7V5IZ 10547590 IC50 > 100000 nM T99932 CIZ1H6 10548866 IC50 = 51000 nM T99932 CRZ8G2 10553070 IC50 > 25000 nM T99932 C08KTS 10570106 IC50 = 39000 nM T99932 CWH0D5 10570570 IC50 = 14000 nM T99932 C3KPO8 10571036 IC50 = 12000 nM T99932 CE4N3P 10572133 IC50 = 15000 nM T99932 C7AHE4 10573618 IC50 = 55000 nM T99932 C8QJH2 10590173 IC50 = 25000 nM T99932 C0YCK7 10591397 IC50 = 33000 nM T99932 CRB09M 10594315 IC50 = 68000 nM T99932 CR0B3N 10595485 IC50 = 60000 nM T99932 C7XQS9 10613843 IC50 > 25000 nM T99932 C12ZAL 10619896 IC50 = 53000 nM T99932 C4XID0 10636108 IC50 = 9000 nM T99932 CKOB90 10639329 IC50 = 5000 nM T99932 C0KFZ3 10640389 IC50 = 21000 nM T99932 C0WS8E 10660380 IC50 = 10000 nM T99932 C3KHD5 10661296 IC50 > 200000 nM T99932 C8UN3P 10663883 IC50 = 100000 nM T99932 CHD97W 10665860 IC50 = 48000 nM T99932 CK0BJ2 10669458 IC50 = 34000 nM T99932 C0PXG8 10683932 IC50 = 10000 nM T99932 C7RK6Y 10685254 IC50 > 25000 nM T99932 C5UIP8 10685991 IC50 > 25000 nM T99932 CW4V3K 10686085 IC50 = 9000 nM T99932 C0S1YO 10687089 IC50 = 89000 nM T99932 CQ5BS6 10688147 IC50 = 20000 nM T99932 CH29QB 10688432 IC50 > 25000 nM T99932 C61YEC 10690566 IC50 = 37000 nM T99932 CZ6S3J 10692755 IC50 > 200000 nM T99932 C49ACR 10694297 IC50 = 13000 nM T99932 CY1JS2 10694592 IC50 = 84000 nM T99932 CFB7U5 10708682 IC50 = 2000 nM T99932 C1GE5N 10712721 IC50 = 16000 nM T99932 C3A9FI 10713603 IC50 > 25000 nM T99932 CVP4S5 10713794 IC50 = 35000 nM T99932 CXP38D 10730172 IC50 > 200000 nM T99932 CEA8F4 10731271 IC50 > 25000 nM T99932 C3EWQ9 10731615 IC50 = 75000 nM T99932 CWS49T 10732591 IC50 > 25000 nM T99932 C5IO6M 10733368 IC50 = 50000 nM T99932 CQ5FM6 10734444 IC50 = 3000 nM T99932 CMN70S 10735519 IC50 = 15000 nM T99932 CWX49K 10736217 IC50 = 5000 nM T99932 C3UG9F 10736883 IC50 = 22000 nM T99932 C1BJ5K 10737740 IC50 > 200000 nM T99932 CRO94K 10740359 IC50 > 25000 nM T99932 CIRT20 10755908 IC50 = 55000 nM T99932 CK2X0E 10756895 IC50 > 100000 nM T99932 C0NL2W 10758494 IC50 = 18000 nM T99932 CTV0Z7 10759371 IC50 = 20000 nM T99932 C71RHU 10762006 IC50 = 9000 nM T99932 C6OD5G 10764262 IC50 = 64000 nM T99932 CKT0A9 10765443 IC50 = 7900 nM T99932 CGVQ48 10779971 IC50 = 12000 nM T99932 C5KY6T 10780887 IC50 > 25000 nM T99932 C41JMB 10782487 IC50 > 200000 nM T99932 CAY0N3 10787769 IC50 > 25000 nM T99932 C28QZK 10803497 IC50 > 100000 nM T99932 CL6RT8 10806631 IC50 = 6000 nM T99932 C3PE6Z 10808807 IC50 = 11000 nM T99932 C1ZOT3 10812014 IC50 = 4700 nM T99932 CM98RG 10826387 IC50 = 5000 nM T99932 CV8SL6 10827468 IC50 = 48000 nM T99932 C2I8UZ 10831571 IC50 = 13000 nM T99932 C5XT1B 10831577 IC50 = 130000 nM T99932 C4Z1VG 10836140 IC50 = 4200 nM T99932 C60MTS 10838771 IC50 > 50000 nM T99932 CZ6AO2 10850191 IC50 > 25000 nM T99932 CQ84TR 10852312 IC50 = 11000 nM T99932 CXT17W 10854252 IC50 > 25000 nM T99932 C7E0YH 10896702 EC50 = 11 nM T99932 CXY64V 11731370 EC50 = 16 nM T99932 C04DFH 11783486 IC50 = 928 nM T99932 C28RVB 11792503 IC50 > 100000 nM T99932 C3VO5H 11824148 IC50 = 1606 nM T99932 CM52YU 14422379 IC50 = 28000 nM T99932 C8USX1 25118615 IC50 = 10000 nM T99932 C94PAD 44382351 IC50 = 25000 nM T99932 CA42ZX 44382442 IC50 > 200000 nM T99932 C8ACR4 44382640 IC50 = 50000 nM T99932 CBI2Y3 44383341 IC50 = 19000 nM T99932 CZB81D 44395506 IC50 = 10.4 nM T99932 CN6E2O 45265215 IC50 = 20000 nM T99932 CBH42D 118711553 IC50 = 20300 nM T99932 C5O8KD 124222736 IC50 = 1200 nM T99932 CE05SO 127038031 IC50 = 15000 nM T99932 C0TOH8 127038032 IC50 = 20000 nM T99932 C70RME 127038387 IC50 = 20000 nM T99932 C2GP1N 127038388 IC50 = 20000 nM T99932 CK5VZ6 127038389 IC50 = 20000 nM T99932 C4G5DV 127038390 IC50 = 20000 nM T99932 C92ENQ 127038391 IC50 = 20000 nM T99932 C0IPO4 127038747 IC50 = 30000 nM T99932 C3CI0D 127038748 IC50 = 30000 nM T99932 C3WCF7 127038749 IC50 = 20000 nM T99932 CS92HL 127039093 IC50 = 40000 nM T99932 C50OZL 127039403 IC50 = 15000 nM T99932 CX14NZ 127041410 IC50 = 10000 nM T99932 C2YG4X 127041411 IC50 > 60000 nM T99932 CW1ZD3 127041716 IC50 = 10000 nM T99932 CEDC62 127041718 IC50 = 20000 nM T99932 CD09BY 127050135 IC50 = 32600 nM T99932 CF2GT1 127051022 IC50 = 20700 nM T99932 CLD3J6 139562057 IC50 = 290 nM T99932 CY95MV 145948918 IC50 = 11900 nM T99932 CN54LI 145960710 IC50 = 2250 nM T99932 CYZW31 145961618 IC50 = 1990 nM T99932 CO5WL0 145961950 IC50 = 2710 nM T99932 C27UMT 145962409 IC50 = 2130 nM T99932 C0UG8V 145962807 IC50 = 4800 nM T99932 CW1OQ2 145963071 IC50 = 2140 nM T99932 C18ECW 145964594 IC50 = 11000 nM T99932 C4VHJ3 145964847 IC50 > 30000 nM T99932 CNT8P1 145965028 IC50 = 6000 nM T99932 CCMN84 145965066 IC50 > 30000 nM T99932 CO4T0U 145965354 IC50 = 9000 nM T99932 CR3YI7 145966075 IC50 = 20000 nM T99932 CFVT97 145966246 IC50 = 30000 nM T99932 CO43ZI 145966328 IC50 = 11000 nM T99932 CQD30F 145966692 IC50 = 20000 nM T99932 C2MEV8 145966854 IC50 = 4000 nM T99932 CI2B6G 145967228 IC50 = 18000 nM T99932 CJDX46 145967246 IC50 = 15000 nM T99932 C98KUB 145967291 IC50 = 20000 nM T99932 CW06TA 145967459 IC50 = 6000 nM T99932 C6L5WA 145969826 IC50 > 30000 nM T99932 C0C6FU 145971874 IC50 = 12000 nM T99932 CKME54 145972363 IC50 = 12000 nM T99932 C0WT5G 145972831 IC50 = 4000 nM T99932 C9PS6E 145973432 IC50 = 300 nM T99932 C9Y2GW 145973540 IC50 = 15000 nM T99932 CWMO63 145974409 IC50 = 500 nM T99932 CP7JG6 145974587 IC50 > 30000 nM T99932 C0A9IQ 145974635 IC50 > 30000 nM T99932 CB84OT 145974761 IC50 > 30000 nM T99932 C8LSE1 145974997 IC50 > 30000 nM T99932 CG0X5M 145976094 IC50 = 11000 nM T99932 CIXO30 145976316 IC50 > 30000 nM T99932 C4VKS2 145976571 IC50 > 30000 nM T99932 CD7KG0 145976625 IC50 > 30000 nM T99932 C0QWS3 145976834 IC50 = 4000 nM T99932 CQ1X3N 145977395 IC50 = 4000 nM T99932 C4B1OR 145977408 IC50 = 7000 nM T99932 CW5E2K 145977530 IC50 = 25000 nM T99932 CHR1E5 145977810 IC50 = 28000 nM T99932 CXR3U7 145977818 IC50 > 30000 nM T99932 CI73TP 145977952 IC50 = 30000 nM T99932 CQN5R6 145977985 IC50 = 8000 nM T99932 C3HUA7 145978193 IC50 = 28000 nM T99932 CP0AQ4 145978399 IC50 = 30000 nM T99932 CHOY97 145978512 IC50 > 30000 nM T99932 CQAY27 145981693 IC50 = 540 nM T99932 CH62WV 145985146 IC50 = 360 nM T99932 D02UYR 9907830 IC50 = 269 nM T99932 D0H2PA 9886977 IC50 = 48 nM T63512 D0P2CS 9409 Ki = 824 nM T63512 D02BGU 76285327 IC50 < 1.7 nM T63512 D07UNH 71543359 IC50 = 2.59 nM T63512 D0NG8Q 75203906 IC50 = 9 nM T63512 CCFH71 11313 IC50 = 1310 nM T63512 CKSE59 17060 Ki = 271 nM T63512 CWZ7F2 22928 IC50 = 18200 nM T63512 C2M7OQ 49561 IC50 = 7800 nM T63512 C9Q7MC 73032 IC50 = 12600 nM T63512 CT98GO 73036 IC50 = 11600 nM T63512 C3VXJ1 74299 IC50 = 3162.28 nM T63512 C6WUO3 102397 IC50 = 37600 nM T63512 C4BO7W 123350 IC50 = 630957.34 nM T63512 C4Z7TA 128167 IC50 = 1644 nM T63512 CX32NQ 171997 IC50 = 18600 nM T63512 C3S5VE 407620 IC50 = 13400 nM T63512 C5V7KY 413246 IC50 = 8900 nM T63512 CAHO89 413248 IC50 = 11600 nM T63512 C6CH0V 413249 IC50 = 1700 nM T63512 CNAS12 414251 IC50 = 8700 nM T63512 CJNR34 414382 IC50 = 13800 nM T63512 C10YZN 414956 IC50 = 19100 nM T63512 CN6WU5 414957 IC50 = 12000 nM T63512 CG6RO4 414958 IC50 = 15500 nM T63512 C0L9MC 415014 IC50 = 9800 nM T63512 CHIZ56 415015 IC50 = 7600 nM T63512 C9ZMT6 416524 IC50 = 5400 nM T63512 CUCH19 595230 IC50 = 794328.23 nM T63512 CW4T8Z 735894 IC50 = 1258925.41 nM T63512 C50KNW 1231279 IC50 = 56 nM T63512 CUD31T 1231283 IC50 > 100000 nM T63512 C0OT5Q 1232321 IC50 = 68 nM T63512 CE16ZI 1232344 IC50 = 111 nM T63512 C5EQ1T 1302891 IC50 = 1200 nM T63512 C9SY6H 1346574 IC50 = 100000 nM T63512 CY7OZ6 1356130 IC50 = 116 nM T63512 C07BCO 1387411 IC50 = 17700 nM T63512 C26EJY 1498816 IC50 > 100000 nM T63512 CHE85D 1517823 Ki = 700 nM T63512 CNA9K3 1808455 IC50 = 5870 nM T63512 CC70QV 1933974 IC50 = 420 nM T63512 C9CV4L 1944172 IC50 = 16100 nM T63512 C1I2XF 2025521 Ki = 5700 nM T63512 CC07UV 2184377 IC50 > 100000 nM T63512 CTQ50F 2195763 IC50 = 2690 nM T63512 CQ4UD0 2263603 Ki = 5000 nM T63512 C8XI0H 2296282 IC50 = 2400 nM T63512 CV1W2Z 2298925 IC50 = 700 nM T63512 CGK89P 2334818 IC50 = 32 nM T63512 CV6X3W 2734359 IC50 = 10000 nM T63512 CL6P5A 2734360 IC50 = 10000 nM T63512 CH3W7A 2734364 IC50 = 5011.87 nM T63512 CB6IN2 2734662 IC50 = 12589.25 nM T63512 C1ZP4W 2763205 IC50 = 1995.26 nM T63512 C15RPB 2773344 IC50 = 5011.87 nM T63512 CO3TB9 2837853 IC50 = 4000 nM T63512 CF21NP 2839033 IC50 = 3700 nM T63512 CM5D4F 2853075 IC50 = 12800 nM T63512 CC8M0K 2854428 IC50 = 3800 nM T63512 C3FDN7 2870670 IC50 = 2200 nM T63512 CN8B3Z 2957873 IC50 = 1500 nM T63512 C4CPR7 3514363 IC50 = 9300 nM T63512 CU1FH7 3585233 Ki = 5800 nM T63512 C3MV8P 3818248 IC50 = 250 nM T63512 C9GQ5C 3933321 IC50 = 261 nM T63512 CND3C4 4672597 IC50 = 10000 nM T63512 CN8XM2 5311263 Ki = 100 nM T63512 C8MGR7 5468154 IC50 = 7400 nM T63512 CR4EP1 5473851 IC50 = 23030 nM T63512 C2VW5J 5507344 IC50 = 1630 nM T63512 CR0M6C 5731347 IC50 = 161 nM T63512 CWM7X8 5793518 Ki = 187 nM T63512 C1GUQ5 5970537 IC50 = 4400 nM T63512 CG15NR 6294465 IC50 = 1584.89 nM T63512 CZO18Y 6484188 IC50 = 251188.64 nM T63512 C4NB1Q 6619710 IC50 = 1242 nM T63512 CQB0F1 7204218 IC50 = 180 nM T63512 CSF81R 7408898 IC50 = 6400 nM T63512 C81MVA 8922263 IC50 = 4900 nM T63512 CGW4B0 8922268 IC50 = 6600 nM T63512 CCS8P0 10110327 IC50 = 6000 nM T63512 CPG04L 10222574 Ki = 200 nM T63512 C69UPR 10225868 IC50 = 220.2 nM T63512 C4ZI8O 11167229 IC50 = 355.6 nM T63512 CFHV74 11568387 IC50 = 597 nM T63512 CFHV37 12527417 IC50 = 300 nM T63512 CH0ZK7 16009052 IC50 = 40 nM T63512 CJF83I 16009163 IC50 = 627 nM T63512 CZO6H5 16045222 IC50 = 727 nM T63512 C2KM0Z 16217683 IC50 = 1000 nM T63512 CQX39H 16217767 IC50 = 316.23 nM T63512 CG73HZ 16218054 IC50 = 501.19 nM T63512 CZ5GY1 20306575 IC50 = 6600 nM T63512 C79EIG 20867282 IC50 = 8811 nM T63512 CFH5B4 20867285 IC50 = 3436 nM T63512 CR29PZ 20867287 IC50 = 29 nM T63512 CGO6S2 20867290 IC50 = 324 nM T63512 C05BUC 23701125 IC50 = 97 nM T63512 CJ5OV6 23701126 IC50 = 120 nM T63512 C9NW0K 24344225 IC50 = 2300 nM T63512 CX30JT 24569174 IC50 = 11400 nM T63512 CMCI21 24882594 Ki = 390 nM T63512 CP13UD 25264721 IC50 = 130 nM T63512 C20SGN 25265312 IC50 = 2.8 nM T63512 C3FO0C 25336524 IC50 = 4100 nM T63512 CBT47L 27825480 IC50 = 8200 nM T63512 CE9QJ8 28431396 Ki < 5000 nM T63512 C7I0CN 32937631 IC50 > 100000 nM T63512 CA3J7Z 32937654 IC50 = 19910 nM T63512 CHVZ30 41539212 IC50 = 4600 nM T63512 CBW7C1 41905902 IC50 = 11400 nM T63512 CH98ME 43608424 Ki < 5000 nM T63512 CA39VQ 44176227 Ki = 367 nM T63512 CPS46Q 44406620 IC50 = 403 nM T63512 CL3FU4 44406630 IC50 = 232 nM T63512 CIX30G 44406632 IC50 = 141 nM T63512 CS28VK 44406644 IC50 = 252 nM T63512 CYUF09 44406648 IC50 = 415 nM T63512 CO1GB3 44406649 IC50 = 803 nM T63512 C7X0EQ 44406669 IC50 = 106 nM T63512 CM57CO 44406671 IC50 = 449 nM T63512 C3ZTC9 44406674 IC50 = 344 nM T63512 C7DY4Q 44406675 IC50 = 238 nM T63512 C91BKR 44406679 IC50 = 363 nM T63512 C5HCR6 44406680 IC50 = 178 nM T63512 CRQB47 44609260 Ki = 3900 nM T63512 CQ62TO 45484131 Ki = 4000 nM T63512 C67BCX 45484132 IC50 = 1500 nM T63512 CO6N1H 45484138 IC50 = 1600 nM T63512 C1WSI0 45484143 IC50 = 16100 nM T63512 C0NL2M 45484148 IC50 = 2500 nM T63512 CZK62B 45484149 IC50 = 17700 nM T63512 C2TS9U 45484156 Ki = 4500 nM T63512 C9Y1PB 45484169 Ki = 7100 nM T63512 C0JR2T 45484172 Ki = 4200 nM T63512 CI90HY 45484179 IC50 = 1300 nM T63512 CDIR60 45484193 IC50 = 5600 nM T63512 C73XEL 45670603 IC50 = 8100 nM T63512 C46NCS 46223667 IC50 = 2410.1 nM T63512 CGT93E 46223902 IC50 = 595.8 nM T63512 C6PNI5 46223904 IC50 = 512 nM T63512 CET63X 46223906 IC50 = 2418 nM T63512 C2YXG1 46230109 IC50 = 1600 nM T63512 CBOC86 46853943 IC50 = 11.9 nM T63512 CLIW46 46853944 IC50 = 29.6 nM T63512 CJ6B4M 46853945 IC50 > 5000 nM T63512 C4LA8P 46855780 IC50 = 2900 nM T63512 CCG89Y 46855781 IC50 = 442 nM T63512 C9P2XE 46855782 IC50 = 13600 nM T63512 C4TQ3B 46855783 IC50 = 2690 nM T63512 CMI9A2 46855784 IC50 > 100000 nM T63512 CEIL64 46855916 IC50 = 60900 nM T63512 CJ63RF 46855917 IC50 > 100000 nM T63512 CW34LA 46856044 IC50 > 100000 nM T63512 C35SNR 46856045 IC50 > 100000 nM T63512 C0HD4K 46856187 IC50 = 2050 nM T63512 CNKA84 46856188 IC50 = 1070 nM T63512 C09TXU 46856189 IC50 = 5.67 nM T63512 CI3J4Z 46856190 IC50 > 5000 nM T63512 CD90ZM 46886463 IC50 = 805 nM T63512 C3O2MW 46911532 IC50 = 28.3 nM T63512 CDL1C3 52458751 IC50 = 4600 nM T63512 C32OLN 52458780 IC50 = 5400 nM T63512 CJ5O0X 53316595 Ki = 4800 nM T63512 C4JZS9 53316596 Ki = 5300 nM T63512 C3PRA9 53316690 Ki = 1600 nM T63512 CWK54O 53317920 Ki = 11000 nM T63512 CX3J6M 53318871 Ki = 3500 nM T63512 CTWQ86 53318947 IC50 = 170.3 nM T63512 C0KF7V 53319248 Ki = 83000 nM T63512 CQ23MZ 53320535 Ki = 26500 nM T63512 CYJ29Z 53320634 Ki = 800 nM T63512 CELI97 53321850 Ki = 1059200 nM T63512 C2GA4O 53323166 Ki = 11100 nM T63512 C87ORL 53323167 Ki = 217500 nM T63512 C82UMS 53323231 Ki = 399000 nM T63512 CAT50B 53324519 Ki = 94 nM T63512 COG70M 53325648 Ki = 22500 nM T63512 CK2XG3 53325837 Ki = 6200 nM T63512 C3XKD0 53361668 IC50 = 5.3 nM T63512 C7X1WA 53361669 IC50 = 6.7 nM T63512 CKG92H 53361670 IC50 = 7.3 nM T63512 CQSG34 53363149 IC50 = 147 nM T63512 C8OFU7 53363236 IC50 = 71 nM T63512 CI9O7S 53363237 IC50 = 10 nM T63512 C39PWF 53363238 IC50 > 5000 nM T63512 CDL3R0 53363240 IC50 = 1594 nM T63512 C7C2WI 53363241 IC50 = 683 nM T63512 CM1B5O 53363330 IC50 = 26 nM T63512 C5GMF7 53363334 IC50 = 59 nM T63512 CH0K9O 55467080 IC50 = 9200 nM T63512 C15CPR 55742744 IC50 = 3400 nM T63512 CF40VE 56666437 IC50 = 8.3 nM T63512 C15KTW 56837805 IC50 = 5 nM T63512 C4ER3Q 56838254 IC50 = 11 nM T63512 CLPQ72 56840629 IC50 > 1000 nM T63512 C9J1ZA 64132279 Ki < 5000 nM T63512 CXMU74 70685363 IC50 = 1200.6 nM T63512 C8HVA2 70685364 IC50 = 1012.8 nM T63512 C02EJB 70691683 IC50 = 361.1 nM T63512 C7AN5L 70693766 IC50 = 704.5 nM T63512 CTB93P 71078085 IC50 < 300 nM T63512 CI51MY 72699322 IC50 = 13 nM T63512 C7HJ4I 73346113 Ki = 800 nM T63512 CD8W6M 73346114 IC50 = 900 nM T63512 CR5TH6 73346115 IC50 = 1000 nM T63512 CAI7F6 73349156 Ki = 200 nM T63512 CA5UP3 73349157 IC50 = 6200 nM T63512 C1WL3E 73353706 IC50 = 1200 nM T63512 C1NWJ9 73355227 Ki = 500 nM T63512 C7SEY9 73355228 IC50 = 1100 nM T63512 CG1XP7 73356770 Ki = 100 nM T63512 C5ZKQ8 73356771 IC50 = 4900 nM T63512 CH6JK3 76284153 IC50 = 86 nM T63512 CN2M8A 76284154 IC50 = 25 nM T63512 C8ZU5I 76284409 IC50 = 206 nM T63512 CZ8W3C 76285000 IC50 = 10 nM T63512 C5ZCG3 76286357 IC50 = 93 nM T63512 C52KTI 76286498 IC50 = 3.5 nM T63512 C0CHU9 78426289 IC50 = 710 nM T63512 C6IB4E 78426290 IC50 = 7609 nM T63512 C3IMC0 78426571 IC50 = 533 nM T63512 CM8B6W 78426572 IC50 = 2021 nM T63512 CDX94E 78426574 IC50 = 246 nM T63512 CTVG49 78427261 IC50 = 12 nM T63512 C1OWG5 78427642 IC50 > 4100 nM T63512 CLPI93 78427773 IC50 = 811 nM T63512 CO7IM8 78428034 IC50 = 1521 nM T63512 C3W7JS 78428035 IC50 = 1708 nM T63512 CRV2I0 78428038 IC50 = 1899 nM T63512 CYA42O 86296259 IC50 < 1.7 nM T63512 CNDS02 86722641 IC50 = 4.2 nM T63512 C89UTJ 86722651 IC50 = 370 nM T63512 CS7T2Z 86722660 IC50 = 150 nM T63512 C3U0PQ 86722669 IC50 = 55 nM T63512 CSG62V 86722720 IC50 = 7.7 nM T63512 CJK6O8 86726538 IC50 = 79 nM T63512 CE7MH9 86726539 IC50 = 4.8 nM T63512 CV6J2P 86726547 IC50 = 10 nM T63512 C9J1YK 90218779 IC50 = 39 nM T63512 CU21YM 90420170 IC50 = 126 nM T63512 CV9HL2 90420193 IC50 = 0.01 nM T63512 C32ZNW 90420330 IC50 = 1001 nM T63512 CKF1O8 90420332 IC50 = 280 nM T63512 CTZY03 90420346 IC50 = 26 nM T63512 C4CD3S 90420388 IC50 = 480 nM T63512 C1X7PZ 90420407 IC50 = 27 nM T63512 CQI95S 90420528 IC50 = 1614 nM T63512 CR3T6L 90420624 IC50 = 103 nM T63512 C97UXT 90420647 IC50 = 261 nM T63512 CK0QF8 90420651 IC50 = 771 nM T63512 C4JQ1N 90420708 IC50 = 122 nM T63512 CX3AU6 90420765 IC50 = 274 nM T63512 CMAH85 90420804 IC50 = 1410 nM T63512 CJ6Q3C 90420931 IC50 = 2372 nM T63512 CI8MB4 90421066 IC50 = 231 nM T63512 CFL32Q 90421072 IC50 = 9163 nM T63512 C8HKB2 90421105 IC50 = 138 nM T63512 C1H6XM 90421207 IC50 = 86 nM T63512 CT6W8B 90421763 IC50 = 1 nM T63512 CZW8O9 90446642 IC50 = 357 nM T63512 C6KHF9 90446729 IC50 = 1684 nM T63512 CZHF20 90446854 IC50 = 2266 nM T63512 CX7SN2 100958879 IC50 > 30000 nM T63512 C5M9IT 101891745 Ki = 71200 nM T63512 CVQG05 117628557 IC50 = 8 nM T63512 CZU05F 117762542 IC50 = 60 nM T63512 CL0IU4 117763631 IC50 = 102 nM T63512 CS29NY 117763635 IC50 = 297 nM T63512 CS03CR 117764297 IC50 = 192 nM T63512 C0IS8Q 117972738 IC50 < 500 nM T63512 CO9P6S 117979336 IC50 = 290 nM T63512 CS8L7E 118631137 IC50 = 30 nM T63512 CZ69HL 118631140 IC50 = 4.2 nM T63512 C13TLC 118705588 Ki = 9 nM T63512 C3QO7C 118705590 Ki = 6.1 nM T63512 CCR7N9 118705591 Ki = 8.1 nM T63512 CY7OB4 118705592 Ki = 18 nM T63512 C8PJ9L 118705594 Ki = 72 nM T63512 CX7PZ6 118705595 Ki = 512 nM T63512 CKY6B7 118705597 Ki = 834 nM T63512 CRWD78 121488120 IC50 = 520 nM T63512 C6JP4Y 121488121 IC50 = 2.5 nM T63512 CI8YL0 122186571 Ki = 2430 nM T63512 CB48IR 122186573 Ki = 3500 nM T63512 CKPY62 122186575 Ki = 1790 nM T63512 CMZQ18 122199235 IC50 = 1 nM T63512 C8LBX9 122445521 IC50 = 5 nM T63512 C7PTS1 122445528 IC50 = 856 nM T63512 CB0OX4 122445531 IC50 = 444 nM T63512 CQT0Y1 122445546 IC50 = 366 nM T63512 CP3OR7 122445549 IC50 = 444 nM T63512 CCHZ25 122445553 IC50 = 68 nM T63512 CCT3I6 122445554 IC50 = 2 nM T63512 C2AP0F 122445559 IC50 = 2 nM T63512 C0SUH4 122445569 IC50 = 3 nM T63512 CQMT18 122445575 IC50 = 2 nM T63512 C95MTN 122445589 IC50 = 3 nM T63512 CX7K1T 122445590 IC50 = 32 nM T63512 CNZ30I 122445606 IC50 = 333 nM T63512 C7KDN0 122445609 IC50 = 10 nM T63512 CZR82Q 122445622 IC50 = 2884 nM T63512 CDXP69 122445627 IC50 = 39 nM T63512 CJ1ZL6 122445633 IC50 = 1060 nM T63512 C4S2BL 122445664 IC50 = 10 nM T63512 CK67WZ 122445670 IC50 = 17 nM T63512 CE37AC 122445741 IC50 = 80 nM T63512 CG08EQ 122445744 IC50 = 2631 nM T63512 CMJH60 122485162 IC50 = 957 nM T63512 CA9K6S 127038370 Ki > 30000 nM T63512 CYTS48 127038371 Ki = 3600 nM T63512 CG08XQ 127038372 Ki > 30000 nM T63512 C5LA4F 127038373 Ki = 1200 nM T63512 C6D2LE 127038374 Ki = 1800 nM T63512 C5F9OI 127038728 Ki < 5000 nM T63512 C16AMS 127038742 Ki = 4000 nM T63512 CF7S4H 127038743 Ki = 3900 nM T63512 C9O0QK 127039698 Ki = 4000 nM T63512 CB2AN6 127041070 Ki > 30000 nM T63512 CI0YJ8 127041071 Ki = 3500 nM T63512 CK4T8G 127041072 Ki = 4500 nM T63512 C45NFG 127041388 Ki > 30000 nM T63512 C2OZH0 127041389 Ki = 1100 nM T63512 CF0CO6 127041685 Ki = 2000 nM T63512 C5C0NZ 127041713 Ki < 5000 nM T63512 CTY79K 127041714 Ki < 5000 nM T63512 C3WOT4 127041715 Ki = 1300 nM T63512 C7R3CT 127045639 IC50 = 170 nM T63512 C8HPR3 127045881 IC50 = 1824 nM T63512 CZ58ER 127045883 IC50 = 13570 nM T63512 CHC46U 129318946 IC50 = 814 nM T63512 C4JIU5 129318948 Ki = 6 nM T63512 C9C6IS 129318949 IC50 = 202 nM T63512 CP3YA0 130272826 IC50 > 10000 nM T63512 CY3P7I 131953432 IC50 = 2.2 nM T63512 CY32UJ 132191122 IC50 = 864 nM T63512 CKO5F8 132191123 IC50 > 1000 nM T63512 CP0SK1 132191124 IC50 = 84 nM T63512 CY2GT4 132191125 IC50 = 18 nM T63512 CIE43Z 132191127 IC50 = 35 nM T63512 CYP6K1 132191129 IC50 > 1000 nM T63512 CVO75D 132191132 IC50 > 1000 nM T63512 C0XQ5V 132191133 IC50 = 190 nM T63512 CS7XL2 132191134 IC50 = 40 nM T63512 CXI92L 132191135 IC50 = 9 nM T63512 CL6K5R 132191136 IC50 > 1000 nM T63512 CZ7EB1 132191138 IC50 > 1000 nM T63512 CS7Y9N 132191139 IC50 > 1000 nM T63512 C74CIN 132191141 IC50 = 70 nM T63512 C6ID7H 132191142 IC50 = 1034 nM T63512 CPQJ60 132191143 IC50 > 1000 nM T63512 CFR76V 132191144 IC50 = 121 nM T63512 CHY9K7 132191145 IC50 > 1000 nM T63512 C1TE6Y 132191148 IC50 = 396 nM T63512 C8U2QW 132191150 IC50 = 98 nM T63512 CY2N3H 132191173 IC50 > 1000 nM T63512 C90OQP 132191174 IC50 = 100 nM T63512 CB0GW7 132191196 IC50 = 67 nM T63512 CA80NH 132191197 IC50 = 56 nM T63512 C49QCS 132191215 IC50 > 1000 nM T63512 CCA8S5 132204178 IC50 > 1000 nM T63512 CR59OC 132204180 IC50 > 1000 nM T63512 C6H5NK 132601734 IC50 = 1800 nM T63512 C8A3OD 132601735 IC50 = 8900 nM T63512 CM5SZ9 134139355 IC50 = 10980 nM T63512 CQC82J 134140698 IC50 = 1252 nM T63512 C6TF7M 134141615 IC50 = 5 nM T63512 CH2IL4 134150544 IC50 = 1251 nM T63512 CWE82P 134153063 IC50 = 2974 nM T63512 CE86OK 134154948 IC50 = 6774 nM T63512 C9ZYQ3 134156757 IC50 = 2430 nM T63512 C1L6HG 135416688 IC50 = 28100 nM T63512 C3CW1E 135422255 IC50 = 17400 nM T63512 CYAZ10 135444386 IC50 = 2420 nM T63512 CN5R2M 135456836 IC50 = 199526.23 nM T63512 CY9D4B 135532641 IC50 = 5900 nM T63512 C5U8GN 136168049 IC50 = 1260 nM T63512 C7Y0HG 137628644 IC50 = 1.23 nM T63512 CHJE20 137633257 IC50 = 258 nM T63512 C0VAH9 137633357 IC50 = 2.99 nM T63512 CPE2B7 137633905 IC50 = 75 nM T63512 CC62IX 137634014 IC50 = 2000 nM T63512 CIK31O 137634199 IC50 > 30000 nM T63512 CFCT50 137634898 IC50 > 30000 nM T63512 CG3JT4 137635448 IC50 > 30000 nM T63512 CFC4B5 137636279 IC50 > 5000 nM T63512 CPFI06 137637376 IC50 > 30000 nM T63512 C8BJY0 137637563 IC50 = 9 nM T63512 C10AQO 137637582 IC50 = 2108 nM T63512 CNSQ34 137637632 IC50 = 10.3 nM T63512 CPJA41 137638308 IC50 > 30000 nM T63512 C7QEC3 137638806 IC50 = 313 nM T63512 CC92YU 137639003 IC50 = 2500 nM T63512 C9C5RW 137639294 IC50 = 75.9 nM T63512 CE2W9H 137639295 IC50 > 30000 nM T63512 CX32KE 137639351 IC50 = 1624 nM T63512 CKF2H4 137639717 IC50 = 563 nM T63512 CS35PR 137639845 IC50 = 4469 nM T63512 C1ZA6R 137640332 IC50 = 5816 nM T63512 CVDE38 137640509 IC50 > 10000 nM T63512 CHBZ25 137640834 IC50 = 25 nM T63512 CLW05V 137641326 IC50 = 5 nM T63512 CW1P4B 137643516 IC50 = 31 nM T63512 CYIL32 137643656 IC50 = 4.47 nM T63512 CU2D1S 137643757 IC50 > 30000 nM T63512 CE2IJ6 137644066 IC50 = 1340 nM T63512 CB5A6R 137644340 IC50 = 25 nM T63512 CZBJ86 137644707 IC50 = 208 nM T63512 C31DFY 137644788 IC50 = 8064 nM T63512 C6YU7C 137644939 IC50 > 30000 nM T63512 C4ZE9K 137645022 IC50 = 204 nM T63512 CK7Q6M 137645163 IC50 > 30000 nM T63512 C4TVJ6 137646414 IC50 = 4246 nM T63512 C9H2DM 137646503 IC50 = 2100 nM T63512 C02VEB 137647488 IC50 = 10568 nM T63512 CX92QL 137647725 IC50 = 30.25 nM T63512 CUP19F 137648170 IC50 > 30000 nM T63512 C64MGY 137648435 IC50 = 493 nM T63512 C4T9PD 137648803 IC50 = 129 nM T63512 C1AX7U 137649756 IC50 = 504.5 nM T63512 CS8QF2 137650111 IC50 = 804 nM T63512 CME95K 137650446 IC50 > 20000 nM T63512 CHU6K8 137650721 IC50 = 1301 nM T63512 C73REU 137650767 IC50 > 100 nM T63512 CT4GH5 137650794 IC50 > 30000 nM T63512 C5ZN6T 137651128 IC50 = 1233 nM T63512 CB3J5U 137651244 IC50 = 660 nM T63512 CE16CD 137651270 IC50 > 8000 nM T63512 C1Y7WH 137652315 IC50 = 10548 nM T63512 C9DPW0 137652437 IC50 > 30000 nM T63512 CD6CP1 137652898 IC50 > 3000 nM T63512 CO85FS 137653791 IC50 = 349 nM T63512 CMX5J8 137654019 IC50 = 500 nM T63512 CGJE10 137654114 IC50 = 1212 nM T63512 C8EK2S 137654233 IC50 = 100 nM T63512 CBN03I 137654401 IC50 > 10000 nM T63512 C3NKE1 137654409 IC50 > 30000 nM T63512 CL9C7W 137655347 IC50 = 2.19 nM T63512 CTI31C 137655405 IC50 = 6570 nM T63512 CJ89KG 137655788 IC50 = 10947 nM T63512 CLH9F4 137656396 IC50 = 11561 nM T63512 C9MP1L 137656859 IC50 = 89 nM T63512 C8YF7V 137656871 IC50 = 2 nM T63512 CI82VH 137657011 IC50 = 63.29 nM T63512 C3J8CF 137658099 IC50 = 1700 nM T63512 C8IN9K 137658724 IC50 > 1000 nM T63512 CPS38V 137658851 IC50 = 9431 nM T63512 CG87RB 137659458 IC50 > 30000 nM T63512 CBC0I7 137659491 IC50 = 717 nM T63512 CQ2X6F 137659539 IC50 > 30000 nM T63512 C9ORD6 137659641 IC50 = 2570 nM T63512 C49HAP 137660293 IC50 = 1000 nM T63512 C2DAE5 137660505 IC50 = 2 nM T63512 CVI8X9 137660570 IC50 > 4000 nM T63512 CJR9T4 137660686 IC50 = 13.67 nM T63512 CI6RL7 137660791 IC50 > 10000 nM T63512 C1Q6SO 137661241 IC50 > 10000 nM T63512 C8FU5H 137661717 IC50 = 1904 nM T63512 C31NLT 145953094 IC50 = 3.9 nM T63512 C9LQ4S 145953763 IC50 = 18 nM T63512 CAN3K8 145960513 IC50 = 170 nM T63512 C7XS0R 145962238 IC50 = 8 nM T63512 C8VXI3 145962560 IC50 = 240 nM T63512 C1JC0O 145963353 IC50 = 10 nM T63512 CKP46R 145963423 IC50 = 1370 nM T63512 CK1VP6 145965172 IC50 = 7.17 nM T63512 CT56CX 145966469 IC50 = 1.75 nM T63512 C5DRB1 145966904 IC50 = 1.79 nM T63512 C5EQ3A 145969591 IC50 = 1.97 nM T63512 CDCL06 145971364 IC50 = 496 nM T63512 COG3E7 145972283 IC50 = 2.78 nM T63512 C4TW2Q 145974696 IC50 = 3.71 nM T63512 C24CIY 145974907 IC50 = 3.29 nM T63512 C12EBM 145975545 IC50 = 8.9 nM T63512 C8HNV1 145975846 IC50 = 5.22 nM T63512 C9W3BA 145976729 IC50 = 4.62 nM T63512 CK1XE5 145976921 IC50 = 7.13 nM T63512 CMJ0O7 145977299 IC50 = 8.44 nM T63512 CX92LS 155511552 IC50 = 3700 nM T63512 C0Z3NP 155511656 IC50 = 2100 nM T63512 C75UDG 155513479 IC50 = 2461 nM T63512 C2EM0L 155514017 IC50 = 5800 nM T63512 C39ZDF 155515348 IC50 = 7500 nM T63512 C7FNT9 155516337 IC50 = 2200 nM T63512 C83ARF 155516516 IC50 = 1070 nM T63512 CEW69G 155518075 IC50 = 8100 nM T63512 C4XTG9 155518368 IC50 = 24 nM T63512 CWT93L 155522727 IC50 = 2.2 nM T63512 C37UGC 155526219 IC50 = 123 nM T63512 CM13PS 155526615 IC50 = 52.3 nM T63512 CUH9K1 155527208 IC50 = 7693 nM T63512 CDKL39 155528817 IC50 = 6200 nM T63512 CB2WI9 155529311 IC50 = 6000 nM T63512 C4HMC0 155530954 IC50 = 23760 nM T63512 CI83LG 155532161 IC50 = 6500 nM T63512 CVX03O 155532639 IC50 = 1600 nM T63512 COF4N6 155536004 IC50 = 19.8 nM T63512 C6M7FZ 155538337 IC50 = 80250 nM T63512 CZ54CX 155538462 IC50 = 2.8 nM T63512 CNQ0V8 155540453 IC50 = 11300 nM T63512 C7V2JR 155542201 IC50 = 5200 nM T63512 C10HXE 155543015 IC50 = 26210 nM T63512 CE16LS 155546544 IC50 = 2200 nM T63512 CIB6H9 155548086 IC50 = 65360 nM T63512 C6V8OJ 155549100 IC50 = 2600 nM T63512 CB8J0V 155549452 IC50 = 1473 nM T63512 C36DRZ 155549655 IC50 = 4600 nM T63512 CP94CR 155549770 IC50 = 5700 nM T63512 C5ASG8 155550687 IC50 = 4 nM T63512 CH2L8M 155551309 IC50 = 4200 nM T63512 C7H0XI 155553495 IC50 = 8900 nM T63512 C28MYP 155559809 IC50 = 7995 nM T63512 CV3X5K 155560593 IC50 = 659 nM T63512 CTL1F7 155561253 IC50 = 6700 nM T63512 CK64JI 155561571 IC50 = 4100 nM T63512 C25AMC 155563065 IC50 = 679 nM T63512 CE1JW7 155564260 IC50 = 27970 nM T63512 CTJK02 155568923 IC50 = 3908 nM T63512 CVTY16 155569460 IC50 = 4944 nM T63512 D01FLQ 2733958 IC50 = 3981.07 nM T63512 D03RKW 9848818 IC50 = 10300 nM T63512 D0A4HS 201262 IC50 = 5011.87 nM T63512 D0AW4G 2734326 IC50 = 5011.87 nM T63512 D0D8OR 2734325 IC50 = 19952.62 nM T63512 D0E1XD 92269 IC50 = 12589.25 nM T63512 D0EJ9B 66827 IC50 = 10000 nM T63512 D0OF2J 24771260 IC50 = 22 nM T63512 D0W6VA 82315 IC50 = 501187.23 nM T63512 D0X7MB 24771259 IC50 = 165 nM T63512 D0ZD6Z 2734370 IC50 = 19952.62 nM T32060 D00TLN 2913 Ki = 0.46 nM T32060 D00XWD 135409453 Ki < 100 nM T32060 D01AZG 5073 Ki = 0.15 nM T32060 D01JMC 11658860 Ki = 1.3 nM T32060 D01UTL 2995 Ki = 160 nM T32060 D01ZII 2726 IC50 = 3.4 nM T32060 D03ELL 2159 Ki = 630.96 nM T32060 D03WEX 9966051 Ki = 180 nM T32060 D04JEE 4946 EC50 > 5011.87 nM T32060 D05XGO 11154555 Ki = 18.8 nM T32060 D05ZIK 4205 Ki = 8.2 nM T32060 D06XZR 27400 Ki = 7.5 nM T32060 D06ZUK 3696 Ki = 94 nM T32060 D07YWY 4417 Ki = 256.45 nM T32060 D08VRO 3822 Ki = 0.23 nM T32060 D09IOI 2170 Ki = 1.77 nM T32060 D0B3UJ 115237 IC50 = 5.2 nM T32060 D0CQ0Z 33630 Ki = 361 nM T32060 D0D1AL 3559 Ki = 25 nM T32060 D0H3HM 60795 Ki = 0.8 nM T32060 D0H7KF 5002 Ki = 31 nM T32060 D0J4JM 5770 Ki > 1000 nM T32060 D0J8JP 10071196 IC50 = 9 nM T32060 D0O6GC 9681 Ki = 10 nM T32060 D0O6SX 3658 Ki = 50 nM T32060 D0P0OU 11978813 Ki = 0.47 nM T32060 D0R1JV 60854 Ki = 0.08 nM T32060 D0R6RO 4184 Ki = 1.2 nM T32060 D0S9MU 5078 IC50 = 7943.28 nM T32060 D0T2XU 4927 IC50 = 23 nM T32060 D0T6QX 5736 Ki = 0.5 nM T32060 D0U2OO 2477 Ki = 851 nM T32060 D0U5OE 3964 Ki = 2.42 nM T32060 D0V4QS 135398745 Ki = 1.585 nM T32060 D0W5HK 216239 Ki = 1959 nM T32060 D0X7DE 4449 Ki = 5.8 nM T32060 D0X7QQ 16363 Ki = 1.2 nM T32060 D0YG7M 3827 Ki = 15.85 nM T32060 D0Z1RV 135398737 Ki = 2.692 nM T32060 D0Z6UC 5358 Ki = 376 nM T32060 D00TLM 6433122 Ki = 0.48 nM T32060 D01IVE 101616 Ki = 7400 nM T32060 D04GMY 11842633 Ki < 100 nM T32060 D08CJK 1150 EC50 = 7.36 nM T32060 D08GJH 125564 Ki = 0.81 nM T32060 D09IRN 21071390 Ki = 791 nM T32060 D0GJ7B 11683556 Ki = 0.51 nM T32060 D0HZ2E 5311271 Ki = 0.1 nM T32060 D0IX1I 123836 Ki = 6.7 nM T32060 D0LI1C 44469321 IC50 > 10000 nM T32060 D0N1HW 5311200 Ki = 200 nM T32060 D0R9HI 11256720 Ki = 26 nM T32060 D0R9KG 11604525 Ki = 4.9 nM T32060 D0U0KR 3035850 Ki > 10000 nM T32060 D0X2XF 177336 Ki < 1000 nM T32060 D0Y6ZK 123683 Ki > 10000 nM T32060 D00PXQ 60785 Ki = 0.04 nM T32060 D01ESB 157918 Ki = 86 nM T32060 D01RAE 133079 Ki > 1600 nM T32060 D02JMI 9888211 Ki = 100 nM T32060 D02VUX 11697676 Ki = 0.14 nM T32060 D02ZSO 6426760 IC50 = 370 nM T32060 D03PJW 108029 IC50 > 1000 nM T32060 D03YPJ 5163 Ki = 1621.81 nM T32060 D03ZZH 9887537 Ki = 251.19 nM T32060 D04DGE 9888804 Ki = 630.96 nM T32060 D05MFO 71781 Ki = 2.455 nM T32060 D06DZI 107780 Ki = 15.85 nM T32060 D08AWI 11430856 Ki > 2000 nM T32060 D0B4BN 3045227 Ki = 31.62 nM T32060 D0B7SP 11292933 Ki = 1000 nM T32060 D0K8NW 5074 Ki = 0.45 nM T32060 D0K9JP 9928332 Ki > 1000 nM T32060 D0M7LV 5761 Ki = 2.6 nM T32060 D0OS6O 60149 Ki = 0.6 nM T32060 D0Q2JS 10436045 Ki = 19.95 nM T32060 D0R5GS 55191 Ki = 3630 nM T32060 D0S5FQ 7153 EC50 = 150 nM T32060 D0T1SF 9909448 Ki = 168 nM T32060 D0U7VZ 11225102 Ki < 100 nM T32060 D0YP7L 6604889 Ki < 5 nM T32060 D0Z7AW 9820261 IC50 = 150 nM T32060 CFJ6H4 1206 Ki = 101000 nM T32060 CZUI83 2769 Ki = 6.31 nM T32060 CP80GT 6088 EC50 = 50.7 nM T32060 CZK5U6 6092 EC50 = 38.3 nM T32060 C7QVM1 8367 EC50 > 10000 nM T32060 C5H9CN 9287 EC50 = 18.9 nM T32060 CFQ7R3 9345 Ki > 10000 nM T32060 C6KIN7 10624 EC50 = 3475 nM T32060 CX96RH 12833 EC50 = 6.27 nM T32060 CHF8L6 12834 EC50 = 8.47 nM T32060 C6Y7RT 15760 EC50 = 6 nM T32060 C6U8OV 16184 Ki = 4.1 nM T32060 CC9A8T 17087 EC50 = 496 nM T32060 CJF27B 17654 EC50 = 2443 nM T32060 CG5T8J 19219 EC50 = 9.02 nM T32060 CJ0C3N 23492 EC50 = 209 nM T32060 CJEV67 26714 EC50 = 44.7 nM T32060 C7VE9O 27557 Ki = 10 nM T32060 CFGH18 27620 Ki = 14 nM T32060 CR69PX 29101 Ki > 10000 nM T32060 C4RF5C 30241 Ki = 2.2 nM T32060 C1LOB9 31014 Ki = 57.9 nM T32060 C8Y6DE 37461 Ki = 2.97 nM T32060 CF3R1X 38240 Ki = 215.6 nM T32060 CGH31L 77158 EC50 = 5.14 nM T32060 COM60X 77379 EC50 = 4.11 nM T32060 C2CG8M 98567 Ki > 10000 nM T32060 C9VZR2 121852 IC50 = 1000 nM T32060 CKP25M 121881 Ki < 1000 nM T32060 CG21YH 127262 Ki = 133 nM T32060 CN92EH 131396 Ki = 8 nM T32060 C4PR2E 132564 Ki = 8.2 nM T32060 C65ECQ 134909 Ki = 5.3 nM T32060 CR5A6M 145709 EC50 = 18.8 nM T32060 CG21LF 154315 Ki = 3 nM T32060 C56XJT 157919 Ki = 86 nM T32060 CV0OJ8 159642 Ki = 397 nM T32060 CLK7P3 169713 IC50 = 6 nM T32060 CF5WT9 171289 Ki > 300000 nM T32060 CX39NY 188249 Ki = 204 nM T32060 CD70NM 190006 EC50 = 75.3 nM T32060 CFH81U 202041 Ki = 112 nM T32060 CVI6X5 213046 Ki = 2 nM T32060 C5NMB6 244378 Ki > 10000 nM T32060 CX7SJ2 334449 IC50 = 35 nM T32060 C68WUF 395901 Ki > 10000 nM T32060 C2V5FA 398712 Ki = 490 nM T32060 CT21SC 411838 Ki = 9530 nM T32060 C0DO9L 417590 Ki = 78 nM T32060 CW9QI0 418242 Ki = 4610 nM T32060 C4O6RK 435595 Ki = 1000 nM T32060 CFJ3R2 452533 Ki > 200 nM T32060 CY1L8V 533915 Ki = 1770 nM T32060 CMT84S 603606 Ki = 676 nM T32060 CU3GF9 606991 Ki = 12000 nM T32060 C17XTV 652557 Ki > 10000 nM T32060 CQW20U 715057 IC50 = 5900 nM T32060 CMIS59 715058 IC50 = 831 nM T32060 C39CWN 728636 EC50 = 1250 nM T32060 CXQ6U0 735755 IC50 > 10000 nM T32060 CZN6S9 743974 EC50 > 39810.72 nM T32060 C2VLP8 752521 Ki = 783 nM T32060 CZ56UF 854024 EC50 = 4.56 nM T32060 CFQ3P0 1078585 Ki = 593.89 nM T32060 CU0H9A 1129292 IC50 = 537 nM T32060 CKG0A5 1158941 Ki = 519.6 nM T32060 C9FI5L 1296368 Ki = 34220 nM T32060 CYE02G 1400243 EC50 < 10000 nM T32060 CGS9R7 2133793 Ki = 29190 nM T32060 CG9N3A 2136365 Ki = 5192 nM T32060 CT8KN9 2232766 Ki = 3905 nM T32060 C0TQ8H 2407992 IC50 = 519 nM T32060 C46RBT 2444416 IC50 = 2130 nM T32060 CX85VC 2581635 Ki > 10000 nM T32060 CA2OY6 2737389 Ki = 1190 nM T32060 C1C4LH 2843443 Ki = 25120 nM T32060 CRA6F5 2853434 Ki = 31530 nM T32060 CL2G3H 2870750 Ki = 6836 nM T32060 CC74QS 2872937 Ki = 33870 nM T32060 CY8R6Q 2948971 Ki = 15830 nM T32060 CV70AM 2989597 Ki = 16 nM T32060 CVD51K 3039995 IC50 = 56 nM T32060 C1FV0B 3045239 Ki = 125.89 nM T32060 C6Z4QI 3050372 Ki = 46 nM T32060 CAM8H3 3066250 IC50 > 1000 nM T32060 C5NA6S 3069135 Ki = 57.6 nM T32060 C4X3VL 3073440 Ki = 421.7 nM T32060 CKB30E 3073449 Ki = 243.22 nM T32060 CAT54M 3074872 Ki = 4677.35 nM T32060 CS5F1I 3083481 Ki = 0.4 nM T32060 CNX8I1 3245407 IC50 = 1500 nM T32060 C69OAZ 3434273 IC50 = 2448 nM T32060 C7YQD3 3519055 Ki > 10000 nM T32060 CS8KE2 3649661 Ki = 174 nM T32060 C0YXV3 3676358 Ki > 10000 nM T32060 CO75SE 3731509 IC50 = 329 nM T32060 C56JID 3763575 Ki = 1.8 nM T32060 CN5YK3 3852202 IC50 = 502 nM T32060 CTH61F 3868902 IC50 > 10000 nM T32060 CXD2W7 3870140 IC50 = 160 nM T32060 CK36GS 3906894 EC50 = 11.75 nM T32060 CB0G8U 4605800 Ki = 0.81 nM T32060 CRUB15 4723431 Ki = 461 nM T32060 C64QUD 5124753 Ki = 0.1 nM T32060 CK8N9Z 5200316 Ki = 105 nM T32060 C83UEY 5234410 Ki = 5.3 nM T32060 CD7U8Z 5311422 Ki < 6309.57 nM T32060 C4J3HP 5640104 Ki = 14960 nM T32060 C4DCR0 5745501 Ki = 79.43 nM T32060 CAO47E 6452095 Ki = 41 nM T32060 CGM63Y 6540428 Ki = 1.585 nM T32060 C0KI9H 6604457 Ki = 153 nM T32060 C3A1FO 6604789 Ki = 12589.25 nM T32060 CC6SM3 6618861 Ki = 125 nM T32060 C0QCK1 6918455 Ki < 2511.89 nM T32060 C1WXY3 6918603 Ki < 2511.89 nM T32060 CD0Z4I 6918648 Ki = 1000 nM T32060 C8AL9V 6918689 Ki = 1445.44 nM T32060 C2VLE0 7048719 Ki = 972.15 nM T32060 CT7GR9 7048721 Ki = 144.54 nM T32060 C2F3BY 7125890 Ki = 10150 nM T32060 CC47WV 9794092 Ki = 18 nM T32060 CXI18K 9794638 EC50 = 269 nM T32060 CCM0S1 9796255 Ki = 1.1 nM T32060 CB5A6I 9799300 Ki < 10000 nM T32060 CE0DI5 9804612 Ki < 10000 nM T32060 C8XGV3 9804849 IC50 = 1900 nM T32060 CNX4F0 9805456 Ki < 2511.89 nM T32060 CZ2WA1 9813163 Ki = 922 nM T32060 CV6LU0 9813187 Ki = 30 nM T32060 C1W2VB 9814248 IC50 = 206 nM T32060 CS1K8O 9814315 Ki = 40 nM T32060 CAD92E 9815159 IC50 = 87.8 nM T32060 C1DT4H 9822580 EC50 = 19 nM T32060 CL38GM 9826580 Ki = 22.9 nM T32060 C38DHN 9834518 Ki = 46 nM T32060 C8AHK9 9834987 IC50 = 179 nM T32060 C1FQ5A 9835490 IC50 = 575 nM T32060 C3W2ZV 9836377 IC50 = 1450 nM T32060 C0H6DZ 9837204 Ki = 217 nM T32060 CWB61S 9838572 Ki = 5.4 nM T32060 CV2A3K 9838959 Ki = 9 nM T32060 CBN06W 9839050 Ki = 2.5 nM T32060 C28HIY 9839057 Ki = 0.04 nM T32060 CWTA61 9839081 Ki = 2.5 nM T32060 CU0HE4 9839392 Ki = 1.8 nM T32060 CYZ47C 9842640 Ki = 770 nM T32060 CWJ75T 9849983 Ki = 60.4 nM T32060 CM13ZV 9856041 Ki = 3.6 nM T32060 C0Q6RX 9856443 Ki = 316 nM T32060 CKQ5O7 9856509 Ki = 10 nM T32060 C9B2QD 9859144 Ki = 32 nM T32060 CRBW42 9861124 IC50 = 206 nM T32060 C0ZR3E 9861687 IC50 = 8128.31 nM T32060 C8M5XK 9863333 Ki = 76 nM T32060 C6ERH9 9863540 Ki > 3000 nM T32060 C0Q6AD 9863611 Ki = 15.85 nM T32060 CI30XR 9865463 Ki = 0.2 nM T32060 C0W3JF 9866423 Ki = 1995.26 nM T32060 C7FBK5 9866660 Ki = 1.175 nM T32060 CSTG23 9866745 IC50 = 107 nM T32060 C57YPX 9867902 IC50 = 5800 nM T32060 C19KGY 9869628 Ki = 398.11 nM T32060 C7AB8O 9870053 Ki < 1258.93 nM T32060 CQ4LC2 9872676 Ki = 583 nM T32060 C86NSR 9877758 Ki = 83 nM T32060 C2ZX0B 9877925 Ki = 2531 nM T32060 CR0EG2 9879772 IC50 = 105 nM T32060 CQJ5X2 9879974 IC50 = 89.5 nM T32060 C2ELZ9 9881053 IC50 = 5000 nM T32060 CKS8Z9 9881119 EC50 = 125 nM T32060 C9NF3D 9881600 Ki = 320 nM T32060 CE46QD 9881885 EC50 = 80 nM T32060 CF59KP 9882393 Ki = 158.49 nM T32060 C10MKO 9882537 Ki = 2.8 nM T32060 CTAC24 9885114 Ki = 1678 nM T32060 CZ8C7G 9885279 Ki = 2.4 nM T32060 C64EOU 9885465 Ki = 0.33 nM T32060 CJW1P5 9888494 Ki = 302 nM T32060 C9GB2M 9888555 Ki = 120 nM T32060 C4PSF6 9888765 Ki = 1.92 nM T32060 C6N8UE 9889681 Ki = 501.19 nM T32060 CM52WU 9890119 Ki = 1000 nM T32060 CEG1K5 9891002 Ki < 1995.26 nM T32060 C7QMK5 9891617 Ki < 1995.26 nM T32060 CEL29O 9891618 Ki = 1000 nM T32060 C6WY0D 9891901 Ki = 679 nM T32060 C3J8GU 9892409 Ki = 630.96 nM T32060 C7EZ8Q 9899243 Ki = 29 nM T32060 C2P3GS 9899500 Ki = 19 nM T32060 CF6OE1 9899545 Ki = 1231 nM T32060 CE28TW 9900179 IC50 = 458 nM T32060 C5TA6D 9903398 Ki = 4.4 nM T32060 CHFP46 9903970 Ki = 0.91 nM T32060 CN3JG8 9904139 Ki = 2884.03 nM T32060 CFI97S 9904205 IC50 = 22.91 nM T32060 CUN81Q 9905249 Ki > 10000 nM T32060 CYWQ50 9906447 Ki = 2718 nM T32060 C7JFZ5 9906978 Ki = 75.8 nM T32060 C2Z9BL 9908431 Ki = 2.6 nM T32060 CYZ5N4 9909089 Ki = 1258.93 nM T32060 CO7BK6 9909648 Ki = 5.8 nM T32060 C78MDV 9913554 Ki = 251.19 nM T32060 C1D4BM 9920585 Ki = 805 nM T32060 CS61ZI 9920667 Ki = 28 nM T32060 C6BTZ9 9920815 Ki = 34 nM T32060 C4BZ3W 9921116 Ki = 1559 nM T32060 CU7JO2 9921840 Ki = 152 nM T32060 CQF2X8 9925089 IC50 = 66.8 nM T32060 CO6MD4 9931534 Ki = 199.53 nM T32060 CXT67L 9931850 IC50 = 12.59 nM T32060 CYVZ47 9934284 Ki = 1995.26 nM T32060 CWO45F 9935387 Ki = 1258.93 nM T32060 CLYE56 9942836 Ki = 199 nM T32060 CS58EO 9944019 IC50 = 379 nM T32060 CX3ZK9 9946374 IC50 = 362 nM T32060 CV1T2W 9947009 IC50 = 787 nM T32060 CH6IJ8 9947172 IC50 = 41.5 nM T32060 CYH3R7 9947817 Ki = 3400 nM T32060 C8T1HO 9948670 Ki = 0.09 nM T32060 CV6M7P 9951882 Ki = 913 nM T32060 C5FJ9S 9951883 Ki = 613 nM T32060 C4YH2I 9953216 Ki = 5.7 nM T32060 CKF9X1 9953268 Ki = 0.52 nM T32060 CK8NR2 9954121 Ki < 3162.28 nM T32060 C3ZQN6 9954930 Ki = 31.62 nM T32060 CFR41N 9957068 Ki < 5011.87 nM T32060 C1NPJ7 9965169 IC50 = 495 nM T32060 C3KTF6 9965610 IC50 = 2010 nM T32060 C6CXJ3 9966330 IC50 = 3180 nM T32060 C0ORJ4 9966331 IC50 = 315 nM T32060 C49MPX 9966437 IC50 = 376 nM T32060 CJ2DK6 9966438 IC50 = 79.4 nM T32060 CC35UV 9966603 IC50 = 301 nM T32060 C36JQD 9970546 Ki = 2.9 nM T32060 CD1IK5 9973432 Ki = 13 nM T32060 C3KLU6 9976913 Ki = 23 nM T32060 CMY73F 9978490 IC50 = 500 nM T32060 CF41ZD 9980157 IC50 = 1932 nM T32060 CC6M7Z 9980998 Ki = 7.2 nM T32060 C76JBU 9981505 Ki < 6309.57 nM T32060 C2PDI5 9982036 Ki = 486.41 nM T32060 C2USG0 9983031 Ki = 158.49 nM T32060 CL9UJ7 9990808 EC50 = 63.1 nM T32060 C9FBE5 9991444 EC50 = 16 nM T32060 C7P2BT 9994008 EC50 = 100 nM T32060 CO0Q6M 9998906 Ki = 16 nM T32060 C98RJC 10000562 Ki = 27 nM T32060 CYG36Z 10003368 Ki < 3162.28 nM T32060 CT2CS3 10003477 Ki < 1000 nM T32060 CQL12P 10004545 Ki > 2000 nM T32060 C3C0YF 10008294 Ki = 1995.26 nM T32060 CLE61D 10015414 EC50 = 42 nM T32060 CS40QN 10015688 Ki = 230 nM T32060 CE3FH2 10015954 Ki < 6309.57 nM T32060 C45HCE 10017554 Ki = 0.48 nM T32060 CEY30Z 10017556 EC50 = 97 nM T32060 C1XK9Y 10019102 IC50 = 6600 nM T32060 CV7R9F 10020040 Ki > 10000 nM T32060 CK18LT 10020895 Ki = 4800 nM T32060 C5X1KG 10022781 Ki = 0.5623 nM T32060 C4KIN3 10024430 Ki = 67.61 nM T32060 C2EUY0 10035109 Ki > 10000 nM T32060 C12LON 10036629 EC50 = 63.1 nM T32060 C2ZO8M 10037962 Ki = 36 nM T32060 C57TZR 10042333 Ki = 1.63 nM T32060 C2C1XS 10042602 Ki = 5.129 nM T32060 C25WVJ 10047566 IC50 > 1000 nM T32060 C6M1TH 10050022 Ki = 794.33 nM T32060 CDSQ03 10058473 Ki = 106 nM T32060 CDKW35 10061837 Ki < 6309.57 nM T32060 C5PG9D 10064386 EC50 = 61 nM T32060 C4PCO3 10065083 Ki = 22 nM T32060 C8Z6MA 10067306 IC50 = 131 nM T32060 CJ50UM 10071897 Ki = 8147.04 nM T32060 C2JFB1 10072280 Ki = 2.5 nM T32060 CKA5F4 10084076 Ki = 469 nM T32060 CD2RM6 10085260 Ki = 13 nM T32060 CJ1RW5 10087864 Ki = 154 nM T32060 CQVJ58 10088453 Ki = 141.25 nM T32060 CVK93I 10090424 Ki = 5.495 nM T32060 C63FME 10090486 Ki = 26.3 nM T32060 CR3D5E 10091430 IC50 = 56.23 nM T32060 CJXQ40 10092819 Ki = 1100 nM T32060 CC5IZ2 10103618 Ki = 98.2 nM T32060 C8F9SD 10105208 EC50 = 100 nM T32060 C7EMN2 10105553 Ki = 60 nM T32060 C54EYD 10108561 IC50 = 389.05 nM T32060 CJ1K5Y 10127939 Ki = 398.11 nM T32060 CZ2S7U 10127968 Ki = 3162.28 nM T32060 C6N2TK 10131545 IC50 = 74.6 nM T32060 CVZ3S9 10132138 IC50 = 249 nM T32060 C26HWK 10132572 IC50 = 1800 nM T32060 CJF76C 10150393 Ki = 2511.89 nM T32060 CI2X3Y 10151289 Ki = 1000 nM T32060 C6FEY0 10151426 Ki = 2.5 nM T32060 C2J8TV 10172764 Ki = 0.39 nM T32060 CP6Q1W 10173403 Ki = 199.53 nM T32060 CN78BA 10176869 Ki = 52 nM T32060 CUJ06B 10194524 Ki > 6309.57 nM T32060 CZB8O2 10198481 Ki = 4.1 nM T32060 C46ECI 10216348 Ki = 4.7 nM T32060 C02TKP 10216639 Ki = 3981.07 nM T32060 CFJY39 10216820 Ki = 125.89 nM T32060 CRNG42 10217207 Ki = 630.96 nM T32060 C96ARE 10217208 Ki = 1584.89 nM T32060 CV1B7C 10217687 Ki = 25.12 nM T32060 CYAV42 10236153 Ki = 4 nM T32060 CRJ01O 10237852 Ki > 1000 nM T32060 CVF1E5 10246054 IC50 = 10.72 nM T32060 CG2B7I 10247701 Ki = 15.14 nM T32060 C2QOD5 10249460 Ki = 15 nM T32060 C4Q2SH 10249573 Ki = 1584.89 nM T32060 C1HT4C 10250754 Ki = 120 nM T32060 C0XJ2W 10250895 Ki = 173.78 nM T32060 CUSP67 10252256 IC50 = 3000 nM T32060 CKT7U9 10254433 Ki = 501.19 nM T32060 CD27VE 10255548 Ki = 125.89 nM T32060 C4BH7J 10256308 Ki = 770 nM T32060 CMRA02 10257042 Ki < 19952.62 nM T32060 CY2KS9 10267283 Ki = 10 nM T32060 CH31DX 10267394 Ki = 232.2 nM T32060 CF2M9O 10268223 IC50 = 36.8 nM T32060 CE9Y8J 10276451 Ki = 17 nM T32060 COAP98 10287912 Ki = 501.19 nM T32060 C9KDO8 10287924 Ki = 3.3 nM T32060 CAT4H3 10288601 Ki > 5011.87 nM T32060 C3WQ8A 10288693 Ki = 4 nM T32060 CPW71K 10309622 Ki = 2511.89 nM T32060 CZVR72 10310067 Ki = 3.5 nM T32060 CU89JD 10314060 Ki = 2311.6 nM T32060 CA3E4W 10316297 Ki = 10.47 nM T32060 CFWC08 10321945 Ki = 398.11 nM T32060 CRT0J7 10329912 EC50 = 1584.89 nM T32060 CE07JM 10330266 Ki = 276 nM T32060 CRH3Z6 10331188 Ki = 65 nM T32060 CT4L5Z 10331841 EC50 = 501.19 nM T32060 CQUG72 10332474 EC50 = 348 nM T32060 CZ60AJ 10333104 Ki = 22 nM T32060 CRQN68 10333842 Ki = 114 nM T32060 C84AVJ 10335309 Ki < 6309.57 nM T32060 CJ4B2X 10335310 Ki < 6309.57 nM T32060 C3E5CB 10337773 Ki = 25118.86 nM T32060 CR3J9S 10338282 Ki = 52.48 nM T32060 CQX86G 10338996 Ki = 3.4 nM T32060 CIQ0G2 10342573 Ki = 0.4 nM T32060 C9IAV3 10346043 Ki > 10000 nM T32060 C86INY 10346749 Ki = 501.19 nM T32060 CS24DU 10353268 Ki = 4.9 nM T32060 CQLD40 10356829 Ki = 6309.57 nM T32060 C0Y4EB 10357163 Ki = 105 nM T32060 CN8PA7 10357986 IC50 > 10000 nM T32060 C32XSA 10358955 Ki = 140 nM T32060 CJR06G 10360487 Ki = 0.3 nM T32060 CM7L5C 10367367 Ki = 0.18 nM T32060 CP43QS 10367835 Ki = 3881.5 nM T32060 CBQ57F 10368126 Ki = 1000 nM T32060 CC1GT2 10368204 Ki = 251.19 nM T32060 CM97GO 10370874 Ki = 6.31 nM T32060 C23KXL 10371119 Ki = 1258.93 nM T32060 C7HCJ3 10379338 Ki = 16 nM T32060 CTWG31 10379339 Ki = 40 nM T32060 CR3KU9 10380133 IC50 > 5000 nM T32060 CDAC63 10381889 IC50 = 3.467 nM T32060 CT78XH 10384138 Ki = 501.19 nM T32060 CO3PZ8 10385090 Ki = 13 nM T32060 CWY94C 10386748 Ki = 114.82 nM T32060 CCK5H3 10388933 IC50 = 79.43 nM T32060 C1R5GY 10390089 Ki < 794.33 nM T32060 C85OHE 10399921 Ki = 13 nM T32060 CA3NO7 10401602 EC50 = 110 nM T32060 C5F4WP 10403711 Ki > 10000 nM T32060 C04WGF 10407367 IC50 = 938 nM T32060 CETH64 10408353 Ki = 58 nM T32060 C0ON1Z 10408409 Ki = 1584.89 nM T32060 C0HSY3 10409174 Ki = 1.479 nM T32060 CYA49X 10409431 Ki < 1258.93 nM T32060 C8S3XE 10409556 IC50 = 48.98 nM T32060 C5PCO9 10410103 Ki < 10000 nM T32060 CSH4O3 10411600 Ki = 27989.81 nM T32060 C9R6GC 10411988 Ki = 4 nM T32060 CK6G0O 10413268 Ki = 316.23 nM T32060 C4TPN1 10413595 Ki > 3981.07 nM T32060 CYMX90 10414272 Ki = 93.2 nM T32060 CUBX84 10420386 Ki = 930 nM T32060 CZ39XA 10424771 Ki = 40 nM T32060 CXVP84 10428830 Ki = 14 nM T32060 C0XZB9 10432760 Ki = 0.28 nM T32060 CD7U5I 10433930 Ki > 10000 nM T32060 CK9QE0 10433973 Ki = 258.23 nM T32060 CY6PV4 10435091 Ki = 0.4 nM T32060 CNJ4Z9 10435572 Ki = 251.19 nM T32060 C2G0AH 10450758 Ki = 16 nM T32060 C8TSH1 10454231 Ki = 1000 nM T32060 C05PSB 10456166 Ki = 31 nM T32060 CA43RM 10457586 Ki < 10000 nM T32060 CSV35T 10458193 Ki = 158.49 nM T32060 C2QO7W 10458785 Ki = 251.19 nM T32060 CTED07 10465263 EC50 = 199.53 nM T32060 C46OBP 10467710 Ki = 160 nM T32060 C2DTK7 10469723 Ki = 30 nM T32060 C5LBS7 10472158 IC50 = 11 nM T32060 CRG9T1 10472780 EC50 = 22 nM T32060 CPI5M7 10476504 Ki = 330 nM T32060 CS01JP 10476876 Ki = 2511.89 nM T32060 CX13YD 10477339 Ki < 5011.87 nM T32060 CEF2O6 10478367 Ki = 6739 nM T32060 CE0CF3 10479090 Ki = 613.76 nM T32060 C12RUZ 10479309 Ki < 1995.26 nM T32060 CH64LD 10479409 Ki = 1258.93 nM T32060 C04TSD 10487869 Ki = 100 nM T32060 CGD21U 10491097 Ki = 5011.87 nM T32060 CB52TQ 10495305 Ki = 0.46 nM T32060 C0CH4G 10495578 Ki = 1995.26 nM T32060 CPG8U3 10495787 Ki = 0.11 nM T32060 C38ZFO 10498110 Ki = 1584.89 nM T32060 CQA0U8 10503674 Ki < 10000 nM T32060 C28FSI 10517019 Ki < 6309.57 nM T32060 CQD7L4 10518435 Ki = 398.11 nM T32060 CUQ03E 10520440 Ki = 0.12 nM T32060 COTM08 10520537 Ki = 6309.57 nM T32060 C2B9PT 10522146 Ki = 0.09 nM T32060 CL1R5C 10523100 Ki = 3162.28 nM T32060 CTO2C7 10526501 Ki = 398.11 nM T32060 CRK20I 10526616 Ki = 100 nM T32060 CNU6K9 10527432 Ki = 251.19 nM T32060 C4EN0P 10528314 Ki = 1000 nM T32060 C3BXP0 10538127 Ki = 398.11 nM T32060 CKG7E2 10541003 Ki = 8500 nM T32060 C4E6TV 10542381 Ki = 0.54 nM T32060 CTCN20 10543551 Ki = 3981.07 nM T32060 CT80DS 10546033 Ki = 63.1 nM T32060 C48BRW 10546334 Ki = 15.14 nM T32060 CV57XZ 10546579 Ki = 0.34 nM T32060 C4S7NI 10549573 Ki = 196.79 nM T32060 CMGY61 10549658 Ki < 10000 nM T32060 CBU41F 10550405 Ki = 5011.87 nM T32060 C0PV1R 10550406 Ki = 501.19 nM T32060 C3P5VL 10550893 IC50 = 35.8 nM T32060 CNB05O 10566712 Ki = 630.96 nM T32060 CMV56C 10567817 Ki = 31.62 nM T32060 C2A6FZ 10568771 Ki = 0.48 nM T32060 CBI9M2 10569827 Ki = 3981.07 nM T32060 C8MSP1 10572269 Ki = 3981.07 nM T32060 C8O0ZN 10573656 Ki = 501.19 nM T32060 C9NQK8 10573762 Ki = 3981.07 nM T32060 CHE80N 10573876 Ki < 5011.87 nM T32060 C4WGZ3 10574607 Ki = 158.49 nM T32060 C09ZXH 10577268 Ki = 50.12 nM T32060 CX8P3I 10583785 Ki = 794.33 nM T32060 CW71RC 10586264 Ki = 125.89 nM T32060 CM97NV 10588666 Ki = 18 nM T32060 CH30OA 10589099 Ki < 6309.57 nM T32060 C8KND3 10589897 Ki = 220 nM T32060 COM18Y 10590891 Ki = 5011.87 nM T32060 CY70EQ 10590892 Ki = 251 nM T32060 C9MUB5 10592633 Ki < 6309.57 nM T32060 C4VLW7 10592646 Ki = 125.89 nM T32060 CH20WS 10593918 Ki < 6309.57 nM T32060 CR1K9O 10594859 Ki = 3981.07 nM T32060 CYNZ23 10595858 Ki = 63 nM T32060 CO23YX 10597140 Ki < 2511.89 nM T32060 C6I3LK 10597210 Ki = 125.89 nM T32060 C2O3BC 10599545 Ki = 1258.93 nM T32060 CAG6B7 10609802 Ki = 335 nM T32060 C74NSJ 10615016 Ki = 4 nM T32060 COM89J 10617682 Ki = 1584.89 nM T32060 CX3A0P 10620719 Ki = 248 nM T32060 CD8KX9 10621491 Ki = 586 nM T32060 CVKA91 10622480 Ki = 79.43 nM T32060 CW8YO5 10623020 Ki < 6309.57 nM T32060 CYT8G2 10623205 Ki = 1584.89 nM T32060 CEWL87 10624604 Ki = 562.34 nM T32060 C0DZC5 10624695 Ki = 1078.95 nM T32060 C8SN9G 10624768 Ki = 5.012 nM T32060 CLCV43 10631592 Ki = 158.49 nM T32060 CQ75TL 10640054 Ki = 2.3 nM T32060 C8C2GN 10640055 Ki = 0.69 nM T32060 CSY57V 10641013 Ki = 158.49 nM T32060 CABG89 10646133 Ki = 251.19 nM T32060 CTJ3V1 10657642 Ki = 60 nM T32060 CE6C0M 10660479 Ki = 1995.26 nM T32060 C38YWE 10670191 Ki = 100 nM T32060 CJC59K 10670813 Ki = 199.53 nM T32060 C4NOI8 10672566 Ki = 181.97 nM T32060 C4BS9A 10673329 Ki = 316.23 nM T32060 C65EDZ 10683685 Ki = 3981.07 nM T32060 CVFC05 10686395 Ki = 2511.89 nM T32060 C9ME8Z 10687130 Ki = 2511.89 nM T32060 CC2I3O 10687827 Ki = 630.96 nM T32060 C7BJO5 10690185 Ki = 1584.89 nM T32060 C2LU1H 10692095 Ki = 220 nM T32060 C7QZO5 10693974 Ki = 251.19 nM T32060 CV7D8G 10696202 Ki = 1009.25 nM T32060 C9GR4O 10696705 Ki = 358.92 nM T32060 CH4X8E 10704473 Ki = 39.81 nM T32060 C7XQN2 10705346 Ki = 398.11 nM T32060 C49IUL 10708935 Ki = 0.43 nM T32060 CML1J4 10709843 Ki = 1258.93 nM T32060 CE8FX4 10709844 Ki = 501.19 nM T32060 C0Y1JL 10710785 Ki = 5011.87 nM T32060 C52SWI 10711404 Ki = 10.2 nM T32060 C7PDA6 10713670 Ki = 0.23 nM T32060 C2SZA0 10714718 Ki = 2511.89 nM T32060 CY3MJ1 10714852 Ki < 6309.57 nM T32060 CJR6Y5 10718089 Ki = 199.53 nM T32060 CJH65T 10738619 Ki = 5011.87 nM T32060 C9F8CO 10739725 Ki = 100 nM T32060 CM3ZH1 10740447 Ki = 501.19 nM T32060 CQ95BN 10740494 Ki = 63.1 nM T32060 CE5U6G 10740495 Ki < 10000 nM T32060 C49CTY 10741816 Ki = 199.53 nM T32060 C8YQE1 10743835 Ki = 5011.87 nM T32060 C7H8VX 10751567 Ki = 368.4 nM T32060 C85XRC 10762125 Ki = 3981.07 nM T32060 C3TD1I 10762475 Ki = 758.58 nM T32060 CAO80C 10762881 Ki = 26 nM T32060 CBUA63 10764263 Ki = 63.1 nM T32060 CQ4X1W 10766449 Ki < 1000 nM T32060 C26JIN 10767350 Ki = 630.96 nM T32060 C5PC0L 10774796 Ki = 100 nM T32060 CK6BG7 10776178 Ki = 70 nM T32060 C3SB0F 10776565 Ki = 125.89 nM T32060 CX0B6M 10781655 Ki = 1258.93 nM T32060 CG9MZ2 10784967 Ki = 2511.89 nM T32060 CF2R3P 10791286 Ki < 1000 nM T32060 C7GF8M 10791443 Ki = 3.981 nM T32060 C8ETQ1 10800216 Ki = 3162.28 nM T32060 CC7J3N 10803066 Ki = 3981.07 nM T32060 CVR74P 10803240 Ki = 398 nM T32060 CEM9Y6 10804534 Ki = 320 nM T32060 CFH1Q4 10805130 Ki = 0.35 nM T32060 CG5B6Z 10808965 Ki = 3162.28 nM T32060 CT65RQ 10811153 Ki = 2511.89 nM T32060 CUD58N 10812577 Ki = 7943.28 nM T32060 CKU7G0 10813396 Ki = 1258.93 nM T32060 CU06IQ 10823155 Ki = 10 nM T32060 CF3N5R 10826203 IC50 = 50 nM T32060 CPXC32 10830245 Ki = 630.96 nM T32060 CCN0A5 10830746 Ki = 1000 nM T32060 C8MHZ9 10835110 Ki < 1000 nM T32060 C5AI2P 10835537 Ki = 1584.89 nM T32060 CFE3J6 10835585 Ki = 5011.87 nM T32060 CGX81B 10837002 Ki = 794.33 nM T32060 CL3XI5 10837468 Ki = 251.19 nM T32060 CCH9T7 10838923 Ki = 1000 nM T32060 CDOH18 10851309 Ki = 10.4 nM T32060 C1R3OJ 10852828 Ki = 5011.87 nM T32060 C0VQ3C 10853014 Ki = 0.25 nM T32060 C62ZSF 10854005 Ki = 63 nM T32060 CV6ZN3 10861900 Ki = 0.42 nM T32060 C20CTE 10873003 Ki = 0.36 nM T32060 CVT7J1 10873805 Ki = 3.62 nM T32060 CRI50E 10885636 IC50 = 715 nM T32060 CB1HY3 10894144 IC50 = 854 nM T32060 CU80EA 10895106 Ki = 220 nM T32060 C5PG3D 10900179 Ki = 6780 nM T32060 CCL2I0 10900237 Ki = 193 nM T32060 CA9XJ5 10905962 Ki = 191 nM T32060 CX65PW 10907460 IC50 = 231 nM T32060 C4SBO9 10915140 IC50 = 460 nM T32060 CO97NK 10921738 Ki = 711 nM T32060 CDR7G5 10925892 Ki = 2.9 nM T32060 C9OI8S 10927262 Ki = 0.66 nM T32060 CU5MZ9 10939073 Ki = 32.1 nM T32060 CGRU15 10969805 Ki = 9.34 nM T32060 C4PK7X 10971209 Ki = 0.41 nM T32060 C5XSE8 10971911 Ki = 227 nM T32060 CK6VF7 10991109 Ki = 9.54 nM T32060 C0BUR1 10991521 Ki = 2.4 nM T32060 C4O7MD 10994400 Ki = 0.91 nM T32060 CJC9K4 11005810 IC50 = 683 nM T32060 C2E8GU 11009992 Ki = 330 nM T32060 CJ4N1Y 11013395 Ki = 970 nM T32060 CE6HJ8 11013863 Ki = 5 nM T32060 C6GT4A 11014340 Ki = 2.692 nM T32060 C3FIP5 11016205 Ki = 1.95 nM T32060 C4T8LY 11020695 Ki = 3.6 nM T32060 CG9JC8 11036563 Ki = 0.53 nM T32060 C01NDT 11036640 Ki = 560 nM T32060 C23JHR 11047568 IC50 = 980 nM T32060 CL5DF2 11057472 Ki = 16 nM T32060 C0SUF4 11057969 Ki = 580 nM T32060 C9ZGU6 11058213 Ki = 15 nM T32060 CG41BK 11071079 IC50 = 1060 nM T32060 CGEY62 11079151 Ki = 31 nM T32060 CS02RN 11085034 Ki = 2300 nM T32060 CL7AX5 11099801 Ki > 2000 nM T32060 CP4WL3 11100243 Ki = 95 nM T32060 C76FKX 11100514 Ki = 3.1 nM T32060 C2YT1Q 11100995 Ki = 150 nM T32060 C7DE0U 11113605 IC50 = 1030 nM T32060 C4HK6I 11120635 Ki = 630 nM T32060 C1HSW0 11123419 Ki > 10000 nM T32060 CHX96W 11133309 Ki = 0.5 nM T32060 CXP12A 11133602 Ki = 130 nM T32060 C73ZDI 11134343 Ki > 10000 nM T32060 C2API9 11141325 Ki = 16 nM T32060 CHEV46 11148641 Ki = 1740 nM T32060 CZK0E6 11150514 Ki > 10000 nM T32060 CTHA45 11151653 EC50 = 53 nM T32060 C18JXF 11153975 Ki = 100 nM T32060 C5HEF8 11154832 Ki = 0.3162 nM T32060 C3NH7G 11160564 EC50 = 125.89 nM T32060 C4SOG5 11163458 Ki = 1070 nM T32060 CW7Y9O 11163741 Ki = 12.59 nM T32060 C8ZN3B 11166042 IC50 = 5168 nM T32060 CK23LI 11166827 Ki = 0.2512 nM T32060 COG98Y 11171955 Ki = 3020 nM T32060 CLP45Z 11175045 Ki = 2620 nM T32060 C75WKP 11176199 IC50 = 20 nM T32060 C6OLX8 11176570 EC50 = 106 nM T32060 C5TR6Q 11178237 Ki = 2.512 nM T32060 C6CL1Y 11178830 Ki = 1995.26 nM T32060 C4FYN6 11185858 Ki > 10000 nM T32060 C0W4SM 11186523 Ki = 1.6 nM T32060 CDA9Z8 11187156 Ki = 627 nM T32060 C90ZAQ 11195293 Ki = 6933 nM T32060 C9N5QU 11200511 Ki = 367 nM T32060 C52BGU 11206703 Ki = 81 nM T32060 C5NA0Z 11209786 EC50 = 513 nM T32060 C41FWO 11213062 Ki = 0.13 nM T32060 C7X9ZC 11221007 Ki = 1700 nM T32060 C2A1PL 11221167 Ki = 59 nM T32060 CAF7T3 11222829 Ki > 10000 nM T32060 CJS0I7 11225281 Ki = 794.33 nM T32060 CA39QR 11227406 IC50 = 920 nM T32060 CZFH27 11231392 Ki = 250 nM T32060 CXB4Q8 11233293 Ki = 2310 nM T32060 CNR71Z 11235362 Ki = 794.33 nM T32060 CBO29U 11236301 Ki = 501.19 nM T32060 C2JOS6 11237290 Ki = 630.96 nM T32060 C9HB3Z 11247569 Ki = 0.5012 nM T32060 C90WSG 11248705 Ki = 3981.07 nM T32060 C3XS7W 11253485 Ki = 1670 nM T32060 C6DA3J 11258838 Ki = 0.5012 nM T32060 CWD43K 11264345 EC50 = 794.33 nM T32060 C92CYH 11265950 Ki = 0.6 nM T32060 C4S2VF 11277147 Ki > 1000 nM T32060 CLFM61 11282335 Ki = 501.19 nM T32060 C28ZWI 11283484 Ki = 0.5012 nM T32060 CJD16T 11288140 Ki > 10000 nM T32060 COQ7H8 11290492 Ki = 3280 nM T32060 C83DSZ 11292350 Ki < 6309.57 nM T32060 C1BHW0 11293856 Ki = 1000 nM T32060 C08UHY 11294575 Ki = 0.2512 nM T32060 C69PBI 11298132 Ki > 10000 nM T32060 CM43ZJ 11300712 Ki = 813 nM T32060 CB0UJ7 11302765 Ki = 431 nM T32060 C9BLC7 11304596 Ki = 794.33 nM T32060 CU4L6M 11304816 IC50 = 2180 nM T32060 C49LMW 11305844 Ki = 251.19 nM T32060 CI79LV 11307899 Ki = 15.85 nM T32060 CLQM72 11312820 Ki > 10000 nM T32060 CU81GW 11313985 EC50 = 47 nM T32060 C1EAK6 11324968 Ki = 260 nM T32060 C46TGM 11328372 Ki < 3981.07 nM T32060 CZ8R4L 11328744 Ki = 0.3162 nM T32060 C2DVE9 11333043 EC50 > 5000 nM T32060 CV1I4W 11336079 Ki = 6560 nM T32060 CKYS02 11336218 Ki = 72 nM T32060 CDN79K 11346775 Ki = 4500 nM T32060 CHW9G0 11347858 Ki = 3050 nM T32060 CC13FL 11349921 IC50 > 10000 nM T32060 CJT5E1 11350623 Ki = 70 nM T32060 CU5L7F 11361103 Ki = 795 nM T32060 C6D1WP 11363880 Ki = 1 nM T32060 CDOP76 11374796 Ki = 0.3162 nM T32060 CBV52J 11384146 Ki = 269 nM T32060 CO1I8H 11384634 Ki = 0.01 nM T32060 CF4OX6 11397149 Ki > 6309.57 nM T32060 C7M3XJ 11397742 Ki = 79.43 nM T32060 C7RAB8 11414184 Ki = 110 nM T32060 COZJ91 11416698 Ki = 1716 nM T32060 CFX98O 11418182 Ki = 0.39 nM T32060 CNM62W 11419526 Ki = 501.19 nM T32060 CIB9K8 11427139 Ki = 829 nM T32060 C7BZA8 11429246 Ki = 0.1585 nM T32060 C3K7TG 11430311 Ki < 1258.93 nM T32060 C4LWN6 11431347 Ki = 0.1995 nM T32060 CYZC62 11437171 EC50 = 111 nM T32060 CF94ZE 11447552 EC50 = 199.53 nM T32060 CY06IJ 11448649 Ki = 67 nM T32060 CHG7Q4 11453346 Ki = 0.2512 nM T32060 CHS2R7 11453704 Ki = 630.96 nM T32060 C1W8QL 11454107 Ki < 1000 nM T32060 CY76VX 11463745 Ki = 1000 nM T32060 CDTI21 11465413 Ki = 398.11 nM T32060 C1QL6G 11475519 Ki = 794.33 nM T32060 CB2X1C 11483068 Ki = 4960 nM T32060 CJ6GV8 11492300 Ki = 7957 nM T32060 CSP63L 11493484 Ki = 157 nM T32060 C8FN2P 11494093 Ki = 83 nM T32060 C9TU8S 11495769 Ki = 0.09 nM T32060 C0AG7D 11497283 Ki = 0.18 nM T32060 CFY18U 11499800 EC50 = 303 nM T32060 CASD80 11501253 Ki = 240 nM T32060 C16AXW 11501537 Ki = 179 nM T32060 CXG04S 11503810 Ki = 2.4 nM T32060 C9BT2W 11512263 Ki = 3.2 nM T32060 CJ2O6D 11514226 Ki = 56 nM T32060 C1TC0B 11517754 Ki = 6.1 nM T32060 CW68BJ 11518143 IC50 = 1000 nM T32060 CT6O8G 11519011 Ki = 0.3162 nM T32060 C9S7ZD 11519589 IC50 = 12.59 nM T32060 C4HI2Q 11531833 Ki = 1 nM T32060 CTA58E 11531941 Ki = 18 nM T32060 C7DBO0 11537385 Ki = 100 nM T32060 CQ08DH 11539632 IC50 = 0.61 nM T32060 C0ZF8J 11544156 Ki = 0.09 nM T32060 CX0DJ3 11545423 Ki = 0.22 nM T32060 C5ZY6N 11545813 Ki = 194.8 nM T32060 C7QKD5 11547151 Ki = 620 nM T32060 CC4J3M 11553617 Ki = 5.1 nM T32060 CW17TM 11554167 Ki = 0.28 nM T32060 C1V5CH 11559090 Ki > 10000 nM T32060 C9UH2M 11559589 Ki = 1.8 nM T32060 CVP1Q9 11567578 Ki = 15 nM T32060 CD3Z7J 11567928 Ki = 33 nM T32060 C3DU6B 11567937 Ki = 0.3162 nM T32060 CNH1K4 11568826 Ki = 180 nM T32060 C5J2UP 11569619 Ki = 7.4 nM T32060 CRK97Z 11570471 Ki = 44 nM T32060 C32JGN 11570589 Ki = 62 nM T32060 C8NMI4 11575479 Ki = 720 nM T32060 CE60FY 11576528 Ki = 140 nM T32060 C4HS8T 11577304 Ki = 6.31 nM T32060 CMTN14 11579853 Ki = 703 nM T32060 C6D1MA 11584660 Ki > 3981.07 nM T32060 CI2FK6 11584858 Ki = 41 nM T32060 C90XFB 11587397 Ki = 1882 nM T32060 C4OK0R 11588889 Ki = 1.259 nM T32060 C1M2CP 11589069 Ki = 17.5 nM T32060 C5TQ3Y 11595191 Ki = 328 nM T32060 CU45DK 11595209 Ki > 10000 nM T32060 CGX8F6 11596869 Ki > 7470000 nM T32060 CVQ4R6 11601955 Ki = 47 nM T32060 C6G7WS 11603119 Ki = 140 nM T32060 CGD62Y 11603486 Ki = 822 nM T32060 C1D5YN 11604671 Ki = 0.3162 nM T32060 CZ2OG1 11608308 EC50 = 125.89 nM T32060 CYF3M8 11609026 Ki = 72 nM T32060 CL51UW 11612277 Ki = 0.6 nM T32060 C9VOB8 11613105 Ki = 93 nM T32060 C5JZ6R 11615459 Ki = 229 nM T32060 C4YG6K 11625339 Ki = 0.2512 nM T32060 CB7M8E 11625642 Ki = 40 nM T32060 CDQ02B 11627746 Ki = 0.28 nM T32060 CN3WL4 11630147 Ki = 1034 nM T32060 C9F4UK 11630623 Ki = 359 nM T32060 C2YHQ0 11633739 Ki = 0.67 nM T32060 C2OU7Y 11638332 Ki > 10000 nM T32060 C19UMY 11638640 Ki = 216 nM T32060 CH89AK 11639248 Ki = 110 nM T32060 C9OXY8 11644842 EC50 > 3000 nM T32060 C9YA0E 11647443 Ki = 0.16 nM T32060 C9XD0H 11649431 Ki = 2.5 nM T32060 CVU40P 11652359 Ki = 6528 nM T32060 CM57PQ 11652452 Ki = 79 nM T32060 C1HDM5 11653679 Ki = 23.6 nM T32060 CPH9X5 11655664 Ki = 15 nM T32060 CRES94 11656729 Ki = 0.3981 nM T32060 CE4FW0 11662306 Ki = 1.6 nM T32060 C4L7TV 11662592 Ki = 1.2 nM T32060 CO2HB4 11663604 Ki = 29 nM T32060 CR7WX0 11665991 Ki = 13560 nM T32060 CI81RY 11666237 Ki = 217 nM T32060 CPR2S8 11668034 Ki = 14 nM T32060 CY0J2U 11670421 Ki = 140 nM T32060 CAI7R5 11673842 Ki = 4441 nM T32060 C7SNQ8 11675550 Ki = 0.631 nM T32060 C4KUL7 11676638 Ki = 4 nM T32060 CMQX39 11676873 Ki = 156 nM T32060 CQZ89L 11684204 IC50 = 0.3981 nM T32060 CEQ6W7 11694810 Ki > 1000 nM T32060 CCE9H2 11695000 EC50 = 10 nM T32060 CDV58J 11696813 Ki = 15.3 nM T32060 CI1LY5 11698617 Ki = 4.5 nM T32060 C2YE9V 11699516 Ki = 150 nM T32060 CU8QZ9 11701315 Ki = 600 nM T32060 CN7Q5B 11710154 IC50 = 1 nM T32060 CRH96P 11716185 Ki = 1488 nM T32060 CV9G1F 11719283 Ki = 0.2512 nM T32060 CB3AM8 11719524 Ki = 1.9 nM T32060 CF3EA1 11719622 Ki = 0.5012 nM T32060 C7T1IL 11720119 Ki = 110 nM T32060 CLYJ75 11729823 Ki = 0.51 nM T32060 C7PVL8 11730467 IC50 = 950 nM T32060 CNH9M5 11733478 Ki = 13.1 nM T32060 C53KHL 11737032 Ki = 586 nM T32060 CH0PB9 11737939 Ki = 383 nM T32060 C05TYZ 11739217 Ki = 3820 nM T32060 C8Q4ET 11742218 Ki = 199.53 nM T32060 CPG15O 11743399 IC50 > 1000 nM T32060 CUE3K5 11749963 Ki < 6309.57 nM T32060 C6SKL1 11750162 Ki = 1258.93 nM T32060 CK4LU1 11750342 Ki < 1000 nM T32060 C45RXA 11750471 IC50 = 0.2512 nM T32060 CT7YB5 11753781 Ki = 501.19 nM T32060 CS68NX 11754336 Ki = 38815.04 nM T32060 C7KD9Z 11766873 Ki = 2511.89 nM T32060 C43JMK 11774776 IC50 = 0.3981 nM T32060 CNZV46 11774955 Ki < 2511.89 nM T32060 C4IQ8G 11775262 Ki = 398.11 nM T32060 CUT31Z 11777150 EC50 = 63 nM T32060 C0CZ2S 11783381 Ki = 3.3 nM T32060 CU5G2Q 11785555 Ki = 5.012 nM T32060 CBM8Q2 11790759 Ki = 296 nM T32060 C09ECB 11792056 Ki = 3162.28 nM T32060 CYZP79 11794624 Ki = 316.23 nM T32060 C6TM2A 11796257 Ki = 199.53 nM T32060 C3U7IY 11797644 IC50 = 2200 nM T32060 C3D2AU 11798958 Ki = 4216.97 nM T32060 C6YZ1Q 11812573 Ki > 10000 nM T32060 CQ98FK 11819486 Ki = 132 nM T32060 CE6J4U 11820166 Ki = 45.9 nM T32060 C4CA7D 11824002 Ki = 1.15 nM T32060 COB43E 11825520 Ki = 1.4 nM T32060 C4CA0B 11826008 Ki = 12.7 nM T32060 CXLW54 11948707 Ki = 2100 nM T32060 CQ64OY 11949706 EC50 = 1428 nM T32060 CP79ZF 11949710 EC50 = 630 nM T32060 CEYG15 11949712 EC50 = 87 nM T32060 CWG8D2 11952353 EC50 = 1500 nM T32060 CK13QD 11953409 IC50 = 5300 nM T32060 C8JQL7 11957735 IC50 > 10000 nM T32060 CR7IZ8 11983273 EC50 = 168 nM T32060 C1QY2P 12005903 Ki = 296 nM T32060 CID7H8 12017581 Ki = 44 nM T32060 CUD9A3 12017598 Ki = 251.19 nM T32060 CM95EO 12017599 Ki = 158.49 nM T32060 C4CE8D 12111141 Ki = 0.06 nM T32060 CL29RB 12197243 Ki = 3 nM T32060 CTMH07 12370465 EC50 = 1399 nM T32060 CL3S9X 12626561 Ki = 0.29 nM T32060 CB4Q6U 12629989 Ki > 10000 nM T32060 CQ4V3A 12737487 Ki = 2542 nM T32060 CJE95C 12898282 Ki = 2073.5 nM T32060 C6I4GL 12901777 Ki = 8540 nM T32060 CL6QH3 12914583 Ki > 10000 nM T32060 C4D6ZV 13059555 Ki = 58.6 nM T32060 C2V9FL 13091268 Ki = 30.9 nM T32060 C2VAE5 13091273 Ki = 12.3 nM T32060 CCG14E 13091356 Ki = 236 nM T32060 C1JW2Q 13091358 Ki = 236 nM T32060 CYN95Z 13091359 Ki = 89 nM T32060 CHO4B1 13547420 Ki = 88.5 nM T32060 CPFQ95 13764011 EC50 = 50.12 nM T32060 CVD25F 13781100 Ki = 94.2 nM T32060 CNW7P2 14248602 Ki = 540 nM T32060 CV08GM 14378574 Ki > 5000 nM T32060 C9I7FG 14515722 Ki > 300000 nM T32060 CBG32N 14515723 Ki = 300000 nM T32060 CGW8C5 14515724 Ki = 100000 nM T32060 C5TU0D 14515725 EC50 = 549.54 nM T32060 C7IXM0 14515726 Ki = 300000 nM T32060 CHIN31 14515727 Ki > 300000 nM T32060 CO8SN6 14515728 Ki > 300000 nM T32060 CSC71V 14555239 Ki = 4490 nM T32060 C6E5IV 14576389 IC50 = 5.2 nM T32060 C4XL7T 14595518 Ki = 1250 nM T32060 C5YF7V 14950933 Ki = 770 nM T32060 CJ16HE 15011385 Ki = 17 nM T32060 CN0KL5 15021875 Ki = 512.86 nM T32060 C5F7NM 15021876 Ki = 1.622 nM T32060 CBQY50 15057516 IC50 = 5.18 nM T32060 C8M4AS 15212884 Ki = 126 nM T32060 C30CHU 15512229 Ki < 316.23 nM T32060 CTPX97 15803947 Ki = 100 nM T32060 CL50KS 15983730 Ki > 5000 nM T32060 C0G2EO 16007117 Ki = 1 nM T32060 C3M8GJ 16026344 Ki = 3866 nM T32060 CLDN43 16046239 Ki = 0.73 nM T32060 C37FIP 16047544 EC50 = 94 nM T32060 C6OYT5 16062136 Ki = 5 nM T32060 CBWZ28 16062137 Ki = 20 nM T32060 CLG47H 16062139 Ki = 11 nM T32060 C6Y3LW 16062143 Ki = 11 nM T32060 C0K1DQ 16062145 Ki = 40 nM T32060 C9HQ7A 16062266 Ki = 13 nM T32060 CM45DK 16062270 Ki = 2.2 nM T32060 C09LXV 16062651 Ki = 29 nM T32060 C8PU1B 16062781 Ki = 13 nM T32060 CCL8Z7 16062782 Ki = 2.5 nM T32060 C7VW3X 16062783 Ki = 11 nM T32060 CXQ0L4 16062784 Ki = 34 nM T32060 CKB71R 16062785 Ki = 4 nM T32060 CPS49Q 16062788 Ki = 0.6 nM T32060 C4AZV6 16062910 Ki = 0.4 nM T32060 CK08NX 16062911 Ki = 0.8 nM T32060 C4JTB1 16062912 Ki = 0.7 nM T32060 CQBU41 16063039 Ki = 8.8 nM T32060 C16OJN 16063047 Ki = 130 nM T32060 C51YGX 16063181 Ki = 9 nM T32060 C3BT8K 16086373 Ki = 15 nM T32060 CGA06C 16086382 Ki = 0.35 nM T32060 CEWI25 16115148 Ki > 10000 nM T32060 CA15XJ 16115267 EC50 = 91 nM T32060 CVL4O8 16115269 Ki = 360 nM T32060 CA15YJ 16115271 Ki = 38 nM T32060 CU86YM 16115381 EC50 = 78 nM T32060 CCZ1E8 16115388 Ki = 91 nM T32060 C3PE9N 16115390 Ki > 10000 nM T32060 C8KMO4 16115392 EC50 > 3000 nM T32060 CIN2U9 16115511 Ki = 2420 nM T32060 CJ1YO5 16115513 Ki = 86 nM T32060 C5RK9P 16115515 Ki = 1473 nM T32060 C4J7OR 16115517 Ki = 43 nM T32060 CVF2A4 16115521 EC50 > 1000 nM T32060 CJO13N 16115644 EC50 = 374 nM T32060 CXNA76 16115647 Ki = 5200 nM T32060 C0F5WY 16115650 Ki = 1040 nM T32060 C4IT3C 16115652 EC50 = 289 nM T32060 CWG94S 16115654 EC50 = 167 nM T32060 C9EF6M 16215237 Ki = 398.11 nM T32060 CNF70V 16220269 IC50 = 15000 nM T32060 CZ2IS9 16660294 Ki > 2207 nM T32060 C6DS7K 16739334 Ki = 1.32 nM T32060 CGCY91 16742745 IC50 = 4580 nM T32060 C2IJ3D 16742746 IC50 = 1810 nM T32060 C4URY2 16742747 IC50 = 8820 nM T32060 CHA74P 16743289 EC50 = 145 nM T32060 C8V1KM 16745235 IC50 = 680 nM T32060 CT9GP4 16763549 Ki = 5264 nM T32060 C0QX5J 17374371 Ki = 18570 nM T32060 C1GR9B 17954204 EC50 = 90 nM T32060 C9WUR7 17956720 Ki = 0.7943 nM T32060 CH31QA 17984294 Ki = 10 nM T32060 C3J2EH 17989823 Ki = 630.96 nM T32060 CV7T6Z 17989828 Ki < 3162.28 nM T32060 CZO18R 17989871 Ki = 630.96 nM T32060 C8JEI2 17989875 Ki < 10000 nM T32060 C9RY6L 18005120 Ki = 251.19 nM T32060 C9PV8A 18180076 IC50 = 1616 nM T32060 CZ58PY 18357723 Ki = 2511.89 nM T32060 C2I7CO 18357724 Ki = 251.19 nM T32060 CS90WO 18357730 Ki = 39.81 nM T32060 CHXQ26 18366015 IC50 > 10000 nM T32060 CK0TX2 18516642 Ki = 100 nM T32060 CNAK30 18715554 EC50 > 1000 nM T32060 CSIT54 18715555 EC50 = 359 nM T32060 CNFG32 18715558 Ki = 230 nM T32060 C03DXY 18715561 Ki = 229 nM T32060 CG2K0J 18715564 Ki = 29 nM T32060 C2ST7K 18735305 Ki = 139 nM T32060 CUC5V9 18735309 Ki = 432 nM T32060 C9GW5T 18735313 Ki = 364 nM T32060 CRLH78 18931123 Ki < 10000 nM T32060 C42WCN 18931133 Ki = 398.11 nM T32060 CW7QF4 18931150 Ki = 125.89 nM T32060 CZKR20 18931163 Ki = 794.33 nM T32060 CW5GP0 18931172 Ki < 10000 nM T32060 C7PU3Q 18931202 Ki = 12.59 nM T32060 C1INB0 18931217 Ki < 10000 nM T32060 CY10RA 18931344 Ki = 3162.28 nM T32060 CODQ12 18931348 Ki = 19.95 nM T32060 C37ZWN 18931357 Ki = 794.33 nM T32060 C5LQX3 18931377 Ki = 1995.26 nM T32060 C5T4BW 18931420 Ki = 1000 nM T32060 CY60VR 18931422 Ki = 1 nM T32060 CQXS12 18986247 Ki = 39.81 nM T32060 CURH72 19036356 Ki = 199.53 nM T32060 C6MQ4P 19036360 Ki = 10 nM T32060 CFB7P2 19036374 Ki = 199.53 nM T32060 CF0X7Z 19036377 Ki = 63.1 nM T32060 C9E0JS 19036385 Ki = 100 nM T32060 C48OSF 19036480 Ki = 31.62 nM T32060 C1HL8Z 19356259 Ki = 251 nM T32060 CJ6L5B 19426632 IC50 = 15.85 nM T32060 C6AOE8 19426635 IC50 = 13.18 nM T32060 CT1Q8M 19426644 IC50 = 25.12 nM T32060 CFYH89 19426650 IC50 > 1000 nM T32060 C9ODM1 19426658 IC50 > 1000 nM T32060 CYFJ81 19926671 IC50 = 1980 nM T32060 C7T8JC 19958494 Ki = 2791 nM T32060 C6LI5E 19958507 Ki = 627 nM T32060 C3M6OA 20026449 EC50 = 7900 nM T32060 C5Q6FW 20576921 Ki = 1.1 nM T32060 C4U8TE 20726100 Ki = 6.5 nM T32060 C71ZTU 20726102 Ki = 12 nM T32060 C5Z7FO 20726104 Ki = 56 nM T32060 CNJY54 20824945 Ki = 22 nM T32060 CSN4T5 20824946 Ki = 290 nM T32060 CRUI61 20824949 Ki = 1100 nM T32060 CBY03N 20846175 Ki < 10000 nM T32060 C9AXD5 20976025 EC50 = 28.1 nM T32060 CPLT36 21044391 Ki = 942 nM T32060 C6JSC0 21044398 Ki = 392 nM T32060 C10IHJ 21073216 Ki = 3.2 nM T32060 CH8EN1 21073533 Ki = 2.9 nM T32060 C1R0SA 21073563 Ki = 0.35 nM T32060 CBUG29 21073579 Ki = 31.2 nM T32060 C15NJA 21073584 Ki = 0.5 nM T32060 CXMG13 21073587 Ki = 12 nM T32060 C57EJD 21073595 Ki = 15.9 nM T32060 CR0D3H 21073606 Ki = 6.7 nM T32060 C60WIT 21073656 Ki = 10.4 nM T32060 C6CQO1 21073658 Ki = 1.5 nM T32060 C1OL3G 21073667 Ki = 1.9 nM T32060 CVT16Y 21073690 Ki = 11.7 nM T32060 C9GHF5 21073716 Ki = 3.3 nM T32060 CA24ZJ 21073731 Ki = 3.5 nM T32060 CGP56E 21073788 Ki = 1.3 nM T32060 C6ARE1 21073793 Ki = 0.19 nM T32060 C3KMW4 21073817 Ki = 50.9 nM T32060 CHM64K 21073872 Ki = 0.79 nM T32060 CAO91K 21099378 Ki = 0.07 nM T32060 C9MDU4 21099413 Ki = 23 nM T32060 C2LMD4 21099424 Ki = 1.43 nM T32060 CJB73F 21099433 Ki = 0.65 nM T32060 CQU60A 21099448 Ki = 28 nM T32060 CBCL34 21099463 Ki = 3.5 nM T32060 C36INC 21099465 Ki = 2.6 nM T32060 C6GRC9 21099470 Ki = 0.7 nM T32060 CY75XP 21099472 Ki = 0.86 nM T32060 CCO7D2 21099473 Ki = 2.6 nM T32060 CP94VE 21099486 Ki = 0.2 nM T32060 CF90PJ 21099505 Ki = 0.65 nM T32060 CDBY94 21099514 Ki = 19 nM T32060 CB12UT 21099515 Ki = 17 nM T32060 CN85CQ 21252889 Ki > 1000 nM T32060 CN1XA4 21252891 Ki > 1000 nM T32060 C6AFN2 21252894 Ki > 1000 nM T32060 CTUY04 21252899 Ki > 1000 nM T32060 C2P1TL 21252902 Ki > 1000 nM T32060 CPWG76 21302447 Ki = 2.8 nM T32060 CQF01H 21302453 Ki = 7.6 nM T32060 CTFH75 21302454 Ki = 79 nM T32060 CGL9D3 21302455 Ki = 70 nM T32060 CY3M2Z 21302456 Ki = 90 nM T32060 CY6H3F 21302457 Ki = 15 nM T32060 CB4V8Q 21302458 Ki = 0.6 nM T32060 C9WD5O 21302459 Ki = 62 nM T32060 C7TSU2 21302471 Ki = 4.2 nM T32060 CWHT46 21302483 Ki = 162 nM T32060 C7Y0HC 21302486 Ki = 0.94 nM T32060 CJP08R 21302487 Ki = 4.7 nM T32060 CB7S2R 21302488 Ki = 2.1 nM T32060 COD3H1 21302489 Ki = 7.5 nM T32060 C2EO0C 21302505 Ki = 2.4 nM T32060 CNP5K6 21439915 Ki = 1810 nM T32060 C3T5HF 21509921 Ki = 23.99 nM T32060 CFN81Q 21527771 Ki = 72 nM T32060 CH59WN 21533446 Ki = 72 nM T32060 C4B0TN 21557475 Ki = 563 nM T32060 CQO1R3 21786603 Ki = 9753 nM T32060 CT7XG9 21830793 Ki = 4975 nM T32060 CSQ2Y0 22017550 Ki = 0.87 nM T32060 C0OIX1 22019270 IC50 = 724 nM T32060 CBN84K 22065997 Ki = 242 nM T32060 CQMS26 22292784 EC50 = 150 nM T32060 C6UXL4 22330705 Ki = 14980 nM T32060 CC6AJ0 22368315 EC50 = 100 nM T32060 CX7F9I 22393282 Ki = 193 nM T32060 CE80BF 22393315 Ki = 2940 nM T32060 CK37OM 22393329 Ki = 2310 nM T32060 C12ICN 22393375 IC50 = 787 nM T32060 C1BL8Z 22393395 Ki = 2235 nM T32060 CX64QZ 22393419 Ki = 224 nM T32060 C3RZ5G 22393430 Ki = 167 nM T32060 CZG9S2 22425072 Ki = 31010 nM T32060 CPD8Q7 22549784 Ki = 28980 nM T32060 C5IE1F 22619858 Ki = 398.11 nM T32060 CD9M5W 22720253 Ki = 136 nM T32060 C9JN0F 22720399 Ki = 82 nM T32060 CB6JH2 22720609 Ki = 45 nM T32060 CNL7Z2 23009084 Ki = 7.2 nM T32060 C2VA8B 23139417 Ki = 1.585 nM T32060 CH5C7X 23288790 Ki = 140 nM T32060 C0NI3J 23290944 Ki = 180 nM T32060 C1RIA7 23395431 EC50 = 100 nM T32060 CA6QL5 23462894 Ki = 400 nM T32060 C0U2TC 23467920 EC50 > 10000 nM T32060 CXD3E6 23625925 Ki = 2.138 nM T32060 CR1M4E 23652278 EC50 = 251.19 nM T32060 CQE1N7 23906630 Ki = 26540 nM T32060 C1A9EF 23983765 Ki = 1.9 nM T32060 CZ4BW9 24044716 IC50 = 161 nM T32060 CFM03J 24208815 IC50 = 670 nM T32060 CQ0KU9 24738459 Ki = 1.83 nM T32060 C0I2HU 24769156 Ki = 66 nM T32060 CGX8K2 24773648 EC50 < 10000 nM T32060 CSCJ40 24773649 EC50 = 10 nM T32060 C6T5XP 24773650 EC50 = 100 nM T32060 CLR9M6 24773651 EC50 = 31.62 nM T32060 CMA8Q6 24773728 EC50 = 316.23 nM T32060 C4O2YA 24773809 EC50 = 125.89 nM T32060 C7IT2S 24773814 EC50 = 251.19 nM T32060 C2U8IH 24773816 EC50 = 100 nM T32060 CTK36B 24773894 EC50 = 2400 nM T32060 CG1V5R 24773895 EC50 = 199.53 nM T32060 C9WV5A 24773897 EC50 = 1000 nM T32060 C6IF2A 24773900 EC50 = 251.19 nM T32060 CNOE28 24773901 EC50 > 5000 nM T32060 C8R9DY 24773978 EC50 = 1584.89 nM T32060 CF2U4K 24773979 EC50 = 1584.89 nM T32060 C2E8SA 24810866 Ki = 18 nM T32060 C14FOH 24810867 Ki = 3.7 nM T32060 CT53OY 24810870 Ki = 3.9 nM T32060 C82ZEQ 24810973 Ki = 9.3 nM T32060 C8GX1Z 24811073 Ki = 408 nM T32060 CX17DO 24811076 Ki = 2470 nM T32060 C6A8SY 24811079 Ki = 6000 nM T32060 CSD96T 24811182 Ki = 865 nM T32060 COQ5U2 24811184 Ki = 3.6 nM T32060 CG0FJ6 24811298 Ki = 18.5 nM T32060 CKCF54 24811301 Ki = 68 nM T32060 C1CH9O 24811415 Ki = 4.5 nM T32060 CG49QZ 24811418 Ki = 36 nM T32060 CGKV62 24811420 Ki = 4.6 nM T32060 CL71GM 24811748 Ki = 4.6 nM T32060 CO6ZG1 24811751 Ki = 270 nM T32060 C5IR4Z 24811854 Ki = 37 nM T32060 C4CU8V 24811856 Ki = 368 nM T32060 CO4ZF3 24811956 Ki = 70 nM T32060 C7RY2Z 24811959 Ki = 1.1 nM T32060 C6IY3J 24812067 Ki = 542 nM T32060 CZL2H0 24812461 Ki = 8.5 nM T32060 CUE6Q0 24812462 Ki = 34 nM T32060 CB6D4T 24812467 Ki = 2.6 nM T32060 CJN09A 24826786 Ki = 326 nM T32060 C3PQB2 24826787 Ki = 84 nM T32060 CRKE01 24826788 Ki = 120 nM T32060 C6BM3J 24826790 EC50 = 64 nM T32060 CF9VK5 24826867 EC50 = 22 nM T32060 CJ7Q4O 24826868 Ki = 85 nM T32060 CT8R9F 24826869 EC50 = 37 nM T32060 C8W9FT 24826870 Ki = 231 nM T32060 CSDP50 24826871 Ki = 511 nM T32060 CGQZ94 24826957 Ki = 146 nM T32060 C5DZ6K 24826963 Ki = 326 nM T32060 C58AMS 24829343 Ki = 19.4 nM T32060 CDC91N 24839550 Ki = 707.95 nM T32060 CY21RE 24841480 Ki = 2400 nM T32060 CBA17N 24849050 EC50 = 116 nM T32060 CUW23K 24854106 Ki = 55 nM T32060 CH2BO5 24861136 Ki = 262 nM T32060 CY18GS 24861188 Ki = 273 nM T32060 C70MST 24861189 Ki = 389 nM T32060 CW1NB6 24861190 Ki = 367 nM T32060 CZ2OX1 24861191 Ki = 110 nM T32060 CA1VQ4 24861192 Ki = 19 nM T32060 C54HEN 24861246 Ki = 222 nM T32060 C2GPJ5 24861249 Ki = 117 nM T32060 CU90ZK 24861250 Ki = 59 nM T32060 CAK91U 24861356 Ki = 89 nM T32060 C3HK0J 24865725 Ki = 2511.89 nM T32060 C0O6FX 24865727 Ki > 6309.57 nM T32060 C98ZIV 24882509 IC50 > 10000 nM T32060 C0KFD3 24884789 Ki = 1584.89 nM T32060 C2NT1L 24887284 Ki = 501.19 nM T32060 C2J0BI 24887285 Ki < 1000 nM T32060 CB41AM 24887289 Ki = 630.96 nM T32060 CC2IJ9 24887290 Ki = 630.96 nM T32060 CXJ90O 24887291 Ki < 5011.87 nM T32060 CTDX79 24887517 Ki = 398.11 nM T32060 C6L7KS 24887518 Ki = 630.96 nM T32060 CPY96D 24887519 Ki = 3981.07 nM T32060 C90ACW 24887525 Ki = 630.96 nM T32060 CR31BN 24887527 Ki = 794.33 nM T32060 C2NVO1 24887761 Ki < 1258.93 nM T32060 C17OXP 24887768 Ki < 3162.28 nM T32060 C24NPA 24887966 Ki < 1584.89 nM T32060 C04UDV 24887967 Ki < 501.19 nM T32060 CHA0N5 24887968 Ki < 1000 nM T32060 CX04AI 24887970 Ki = 794.33 nM T32060 C0DX5I 24888180 Ki = 630.96 nM T32060 CO74UR 24888181 Ki = 398.11 nM T32060 CGLH34 24888182 Ki < 2511.89 nM T32060 C6R9EH 24888183 Ki = 630.96 nM T32060 CZX93A 24888184 Ki < 1000 nM T32060 C1GR0V 24888185 Ki = 398.11 nM T32060 CZY2P8 24889531 Ki = 1.8 nM T32060 CAOF91 24894071 IC50 > 1000 nM T32060 C69AYD 24900557 Ki = 2.399 nM T32060 C4IGH9 24936042 Ki = 1100 nM T32060 CW4X0E 24962988 EC50 > 10000 nM T32060 CA20NZ 25025581 Ki = 158.49 nM T32060 C6DO4B 25032525 Ki = 0.33 nM T32060 C7O8YH 25068794 Ki = 1.76 nM T32060 CZ9SN8 25068797 Ki = 0.72 nM T32060 CL46IP 25068850 Ki = 5.07 nM T32060 CEH7D9 25068903 Ki = 0.483 nM T32060 CB03DL 25068905 Ki = 14.9 nM T32060 C5ZHN9 25068906 Ki = 3.37 nM T32060 C0ZJB7 25068907 Ki = 11.3 nM T32060 C9G7EM 25068908 Ki = 3.54 nM T32060 CZBY61 25068962 Ki = 11.1 nM T32060 CP9G5Z 25068963 Ki = 4.86 nM T32060 CB3F0I 25068964 Ki = 3.16 nM T32060 CCO7B3 25068966 Ki = 4.29 nM T32060 C16ERI 25069015 Ki = 20.1 nM T32060 CZM94A 25069016 Ki = 25.3 nM T32060 CYZ45N 25069072 Ki = 11.2 nM T32060 CEB96S 25069073 Ki = 3.35 nM T32060 CAI7V1 25069074 Ki = 5.44 nM T32060 C8A3HM 25069121 Ki = 10.1 nM T32060 CG5WX6 25069122 Ki = 126 nM T32060 CS8VK1 25069125 Ki = 53.4 nM T32060 CHZB81 25069180 Ki = 7.91 nM T32060 C3W1AX 25069181 Ki = 17.1 nM T32060 CPGZ03 25069239 Ki = 32.1 nM T32060 CT0R3H 25069240 Ki = 2.68 nM T32060 CX5JF4 25069241 Ki = 1.19 nM T32060 C1P4EC 25069242 Ki = 38.5 nM T32060 CCV27I 25069243 Ki = 13 nM T32060 C5BR0K 25069297 Ki = 10 nM T32060 CU34CX 25069298 Ki = 3.49 nM T32060 C0Z6YL 25069299 Ki = 13.8 nM T32060 C5Z9MA 25069300 Ki = 2.21 nM T32060 C1OGS2 25069301 Ki = 0.904 nM T32060 C53LJG 25069302 Ki = 3.45 nM T32060 CX74UK 25069353 Ki = 5.41 nM T32060 C8F6VC 25069354 Ki = 1.08 nM T32060 C56RCY 25069355 Ki = 2.1 nM T32060 CI7SM5 25069356 Ki = 3.07 nM T32060 C4B0FU 25070577 IC50 = 119 nM T32060 CBY3O2 25070582 EC50 = 68 nM T32060 CI8NL3 25071384 Ki = 240 nM T32060 C6F5SU 25071385 Ki = 350 nM T32060 CL7TN4 25071691 Ki = 4 nM T32060 C75ZIC 25071692 Ki = 490 nM T32060 C49ZFU 25072002 Ki = 110 nM T32060 C8OBV4 25072633 Ki = 210 nM T32060 CS1CI4 25072941 Ki = 1500 nM T32060 C9SZG1 25084025 EC50 = 1680 nM T32060 CBKG34 25093832 Ki = 91 nM T32060 C2YJX3 25099159 Ki = 8.318 nM T32060 CMX36H 25107505 Ki > 7710 nM T32060 CR17NY 25110703 Ki = 25.12 nM T32060 CJK06X 25110705 Ki = 43 nM T32060 CTV61A 25110708 Ki = 375 nM T32060 CVIB80 25110709 Ki = 121 nM T32060 CA1EJ2 25120700 IC50 = 5800 nM T32060 C2FY7C 25128757 Ki = 70.1 nM T32060 C5NW4M 25129807 Ki = 4770 nM T32060 CQKP18 25130148 Ki = 2.512 nM T32060 CAV81B 25130157 Ki = 171 nM T32060 C7TQ4B 25130505 Ki = 17.38 nM T32060 CD04PQ 25130829 Ki = 1.549 nM T32060 CM58BO 25130830 Ki = 6.918 nM T32060 C9HYT3 25130831 Ki = 1318.26 nM T32060 C36NMK 25130836 Ki = 5.129 nM T32060 C1MNU0 25131483 Ki = 25.7 nM T32060 CZ6NK0 25131829 Ki = 21.88 nM T32060 C67QCG 25132869 Ki = 2800 nM T32060 CV0TM5 25138698 Ki = 3.2 nM T32060 C5B4LT 25138700 Ki = 43 nM T32060 CH7DR0 25138857 Ki = 200 nM T32060 CGBL04 25139014 Ki = 1.3 nM T32060 CIUX26 25139019 Ki = 3.5 nM T32060 CJ5VX0 25140466 Ki = 7 nM T32060 CI3OM1 25140468 Ki = 23 nM T32060 CGON30 25140471 Ki = 107 nM T32060 CL84YJ 25141534 Ki = 48 nM T32060 C5C7GH 25184832 Ki = 31.62 nM T32060 C6ZY3B 25186020 Ki = 300 nM T32060 CN06PX 25209050 Ki = 19.95 nM T32060 CR1K8B 25209356 Ki = 2951.21 nM T32060 CLKT16 25209357 Ki > 7413.1 nM T32060 CDF83Q 25209705 Ki = 6.31 nM T32060 C6PL1Y 25256817 Ki = 10 nM T32060 C15QMB 25263320 IC50 > 1000 nM T32060 C2QLS7 25375331 Ki = 1784 nM T32060 CRB9W7 25450664 Ki > 10000 nM T32060 C8FWE5 25456694 Ki > 10000 nM T32060 CEK31Q 25487292 Ki = 2033 nM T32060 CN39GC 25491778 Ki > 10000 nM T32060 C1QT2Y 28071610 Ki = 4554 nM T32060 CU9PY2 28357663 Ki = 334 nM T32060 CYKH58 28390601 Ki = 53 nM T32060 C1D2LR 29943048 Ki = 2.6 nM T32060 CMT4F6 30859353 IC50 = 24.2 nM T32060 CN0JB7 30859354 IC50 = 1378 nM T32060 CA93TJ 30859359 IC50 = 2618 nM T32060 CEZ1A6 32718395 Ki = 3430 nM T32060 C9QGK3 34257212 Ki = 17 nM T32060 CA58DL 41305446 Ki = 6794 nM T32060 CG56DF 42388639 IC50 = 85 nM T32060 CH5QX6 42389467 IC50 = 74 nM T32060 CCYP13 42605775 Ki = 5 nM T32060 CKH3P1 42606928 Ki = 1.6 nM T32060 CZ80TE 42607158 IC50 = 4 nM T32060 CQS4M3 42607276 Ki = 3.6 nM T32060 CUS06A 42629118 Ki = 2100 nM T32060 CY7W2J 42631003 Ki = 1.2 nM T32060 CV2X5B 42635027 IC50 = 352 nM T32060 CS9Q3H 42635204 IC50 = 95 nM T32060 CQ2M5S 42635387 IC50 = 19 nM T32060 CR3KM7 42635388 IC50 = 1824 nM T32060 CJ3NP5 42636941 IC50 > 10000 nM T32060 C0AI7N 43229249 Ki = 3.89 nM T32060 CK0C3Z 43282996 IC50 = 1050 nM T32060 C2VNA3 43283055 IC50 = 66.4 nM T32060 CP16RL 43285101 IC50 = 55.1 nM T32060 C0VC7J 43314210 IC50 = 52.4 nM T32060 CYV94L 43314375 IC50 = 274 nM T32060 C9QJ4Z 43386604 IC50 > 10000 nM T32060 CJ41QV 44126269 Ki = 1.096 nM T32060 CMR7T1 44204999 Ki = 3.162 nM T32060 CVG6X1 44209472 Ki = 18 nM T32060 CD5AB7 44209480 Ki = 50 nM T32060 CQ8NV3 44214723 Ki = 398.11 nM T32060 CSVN47 44214724 Ki = 316.23 nM T32060 CJ8F5Y 44215629 Ki = 30 nM T32060 CT29ZS 44216196 Ki = 2.7 nM T32060 CRNL71 44225654 EC50 = 32 nM T32060 CH59RP 44247803 Ki = 0.14 nM T32060 C2FDB1 44250364 IC50 > 1000 nM T32060 C8MC0Q 44251387 IC50 > 1000 nM T32060 C5YEA8 44251388 IC50 > 10000 nM T32060 C0BSF6 44251389 IC50 > 10000 nM T32060 C2K0VZ 44253016 Ki > 2511.89 nM T32060 C83XZI 44264336 Ki = 1300 nM T32060 CKP90T 44265170 Ki = 2.5 nM T32060 C6FZ5D 44265202 Ki > 50000 nM T32060 C5HP8Z 44265227 Ki = 10 nM T32060 CP8S2J 44266156 Ki = 31.62 nM T32060 CM0CW8 44266160 Ki = 42.66 nM T32060 C0P8IF 44266163 Ki = 1.698 nM T32060 CU67NF 44266164 Ki = 186.21 nM T32060 C14ACY 44266178 Ki = 223.87 nM T32060 CN3ES2 44266182 Ki = 48.98 nM T32060 CKLS45 44266203 Ki = 269.15 nM T32060 CARU58 44266221 Ki = 6.918 nM T32060 CA1WJ4 44266222 Ki = 19.5 nM T32060 CS2MU8 44266229 Ki = 154.88 nM T32060 CZ84XC 44266244 Ki = 54.95 nM T32060 CR16DY 44266245 Ki = 74.13 nM T32060 CVHM20 44266253 Ki = 977.24 nM T32060 C1FTY0 44266268 Ki = 16.98 nM T32060 C0C6RL 44266289 Ki < 1584.89 nM T32060 C5NS9O 44266315 Ki = 77.62 nM T32060 CCP37Q 44267158 IC50 = 10000 nM T32060 CFEI56 44267161 IC50 = 7762.47 nM T32060 CHU4L9 44267168 IC50 = 11220.18 nM T32060 CIZ5W7 44267181 IC50 = 15848.93 nM T32060 CFE12G 44267205 IC50 = 24547.09 nM T32060 C5CPZ7 44267215 IC50 = 213796.21 nM T32060 C7Z4RE 44275982 Ki > 10000 nM T32060 CU35RG 44276349 Ki > 10000 nM T32060 CC2OD4 44278111 Ki = 1932 nM T32060 CRMA84 44278114 Ki > 10000 nM T32060 CF0Y4M 44278115 Ki = 509 nM T32060 CGBY51 44287166 Ki > 10000 nM T32060 C85DJE 44287175 Ki = 38 nM T32060 C0LGX2 44287190 Ki = 230 nM T32060 C2GB5A 44287459 Ki = 4300 nM T32060 C8EY2C 44289762 Ki = 178 nM T32060 COS7M9 44289763 Ki = 2355 nM T32060 CHM25N 44290039 Ki = 1350 nM T32060 C7HTM5 44290348 Ki > 10000 nM T32060 CG62JB 44298021 Ki = 794.33 nM T32060 CV5YP3 44298022 Ki = 158.49 nM T32060 CY1B3H 44298079 Ki > 10000 nM T32060 CCU89I 44298080 Ki = 100 nM T32060 C9TS2N 44298082 Ki = 158.49 nM T32060 CY0VX7 44298086 Ki = 63.1 nM T32060 CSIC31 44298091 Ki = 501 nM T32060 CZ7BV3 44298092 Ki > 794.33 nM T32060 CO06KG 44298100 Ki = 3162.28 nM T32060 C1AF0K 44298108 Ki > 794.33 nM T32060 C9AVQ8 44298118 Ki = 1995.26 nM T32060 C6Z0QR 44298120 Ki > 1000 nM T32060 C41MRW 44298121 Ki = 1000 nM T32060 CP0D3F 44298126 Ki > 10000 nM T32060 C3KUI9 44298129 Ki > 10000 nM T32060 CH2UE9 44298138 Ki = 100 nM T32060 CPL7S5 44298140 Ki = 158.49 nM T32060 CJ3H6P 44298142 Ki = 316 nM T32060 C1SBI3 44298147 Ki > 10000 nM T32060 CI9S7T 44298151 Ki > 5011.87 nM T32060 CUQ5J7 44298157 Ki > 6309.57 nM T32060 CV14AJ 44298158 Ki = 5011.87 nM T32060 CG46JN 44298163 Ki = 15.85 nM T32060 CE8C1H 44298172 Ki = 79.43 nM T32060 CS6XN2 44298173 Ki = 7.943 nM T32060 CO9YU5 44298175 Ki = 100 nM T32060 C93TDS 44298176 Ki = 79.43 nM T32060 CIP20E 44298182 Ki = 3981 nM T32060 C5EDF3 44298186 Ki = 630.96 nM T32060 C71ZLS 44298192 Ki = 1584.89 nM T32060 C0IC9T 44298193 Ki > 10000 nM T32060 CX64BM 44298208 Ki = 630.96 nM T32060 CF1K0H 44298209 Ki > 630.96 nM T32060 C7L1FM 44298225 Ki = 501.19 nM T32060 C3NK6M 44298226 Ki = 794.33 nM T32060 CU0FL2 44298229 Ki = 125.89 nM T32060 CE1Y5J 44298230 Ki = 125.89 nM T32060 C0N3KH 44298234 Ki = 251.19 nM T32060 C9YRS1 44298236 Ki = 125.89 nM T32060 C14RQX 44298243 Ki = 158.49 nM T32060 CWC4O2 44298244 Ki = 158.49 nM T32060 C58LBP 44298246 Ki = 251.19 nM T32060 CX2WP8 44298249 Ki > 794.33 nM T32060 C2Q5ZP 44298254 Ki = 501.19 nM T32060 CKY68S 44309775 Ki = 330 nM T32060 C1TKV6 44309876 Ki > 10000 nM T32060 CI8XJ3 44312903 Ki = 99 nM T32060 C65ARQ 44313164 Ki = 110 nM T32060 CK5WM1 44313266 Ki = 52 nM T32060 CO0X8D 44315397 Ki = 440 nM T32060 CWH8V9 44315398 Ki = 32 nM T32060 CP0C2G 44315697 Ki = 58 nM T32060 C7VS1O 44315715 Ki = 233 nM T32060 C6QD8K 44315716 Ki = 116 nM T32060 CNSW85 44315725 Ki = 70 nM T32060 CUJP95 44315801 Ki = 1581 nM T32060 CRI0J2 44315943 Ki = 426 nM T32060 CALI20 44315965 Ki = 146 nM T32060 CW0P1Z 44315966 Ki = 141 nM T32060 CF40WU 44315993 EC50 = 164 nM T32060 CD30XR 44315994 Ki = 88 nM T32060 COW64J 44315995 Ki = 182 nM T32060 C1GQT9 44316017 Ki = 167 nM T32060 CG5P9D 44316018 Ki = 102 nM T32060 CS25VN 44316027 Ki = 184 nM T32060 CQTB64 44316053 Ki = 756 nM T32060 CQ50LG 44316215 Ki > 10000 nM T32060 C1L3DB 44318442 IC50 > 1000 nM T32060 CV8WZ0 44318454 IC50 = 1.148 nM T32060 CMQW13 44318461 IC50 = 91.2 nM T32060 CPIT23 44318554 IC50 = 23.99 nM T32060 C75CNK 44318581 IC50 = 6.918 nM T32060 C84MTV 44318695 IC50 = 22.39 nM T32060 C8LK5W 44318820 IC50 = 10.47 nM T32060 C35OHA 44318834 IC50 = 32.36 nM T32060 CWN39R 44318841 IC50 = 47.86 nM T32060 CXJL56 44318842 IC50 = 3.09 nM T32060 C7CTF9 44318853 IC50 > 1000 nM T32060 CM39LE 44319098 IC50 = 1000 nM T32060 C5NG8E 44319099 IC50 > 1000 nM T32060 C3RV7M 44319119 IC50 = 302 nM T32060 CY8L5E 44319120 IC50 = 31.62 nM T32060 CE0I4R 44319133 IC50 = 53.7 nM T32060 C9MY2X 44319134 IC50 = 67.61 nM T32060 CHT83A 44320347 Ki = 14 nM T32060 CEA13Y 44323840 Ki < 10000 nM T32060 CNYT01 44323874 Ki = 0.3 nM T32060 CPB89X 44323908 Ki < 10000 nM T32060 C3MXG7 44324011 Ki < 10000 nM T32060 C4KGL6 44324017 Ki = 0.14 nM T32060 C2MSG8 44324041 Ki = 0.14 nM T32060 CY03UK 44324042 Ki = 0.08 nM T32060 C5IFM9 44324046 Ki = 0.43 nM T32060 CE3BO7 44324047 Ki = 2.6 nM T32060 C3C5LO 44324051 Ki = 0.19 nM T32060 C1NFW3 44324052 Ki = 0.13 nM T32060 C2W0VB 44324056 Ki = 3.5 nM T32060 CT48CS 44324065 Ki = 0.26 nM T32060 C9UR6K 44324070 Ki = 1.7 nM T32060 CO25PJ 44324071 Ki > 1000 nM T32060 CPZ7N8 44324079 Ki = 4 nM T32060 CF72QK 44324084 Ki = 3000 nM T32060 CM45XW 44324091 Ki = 0.18 nM T32060 CGOY42 44324142 Ki = 6.31 nM T32060 CFG52Q 44324224 Ki = 1.2 nM T32060 CLKI67 44324247 Ki = 7.3 nM T32060 CW16JD 44324737 Ki > 1000 nM T32060 CA84SN 44324765 Ki > 1000 nM T32060 COA3H4 44324800 Ki > 1000 nM T32060 CY04JW 44324972 Ki > 1000 nM T32060 C29NRF 44326124 Ki = 68.7 nM T32060 CHR3P2 44326125 Ki = 433 nM T32060 C0C1LX 44326219 Ki = 56 nM T32060 CTC70Y 44326298 Ki = 102 nM T32060 C2OZT8 44326319 Ki = 21.7 nM T32060 C8TQL9 44326320 Ki = 92.6 nM T32060 C0GJ3W 44326321 Ki = 37 nM T32060 CUJ74H 44326336 Ki = 30.7 nM T32060 CGE89D 44326357 Ki = 80.7 nM T32060 C3VT2B 44326358 Ki = 90.5 nM T32060 C3A1WX 44326390 Ki = 433 nM T32060 C9KA7Y 44326405 Ki = 1064 nM T32060 CCSV14 44326407 Ki = 86.5 nM T32060 CY4C9X 44326422 Ki = 48.6 nM T32060 CTGR29 44326427 Ki = 433 nM T32060 CKHM97 44326433 Ki = 1088 nM T32060 CIC4V1 44326442 Ki = 17.3 nM T32060 CW2A8X 44326690 Ki = 104 nM T32060 C5HW0O 44326705 Ki = 19.6 nM T32060 C4AI2N 44335528 Ki = 69.9 nM T32060 CV19HU 44335657 Ki = 61.1 nM T32060 CRS9N1 44335683 Ki = 5.7 nM T32060 CK4I9F 44335687 Ki = 4.3 nM T32060 CM58WP 44335695 Ki = 11.5 nM T32060 CV9G7R 44335697 Ki = 11.8 nM T32060 CKRQ49 44335713 Ki = 22.8 nM T32060 CQ3P6N 44335719 Ki = 12.5 nM T32060 CXA43J 44335732 Ki = 18.3 nM T32060 COAV62 44335766 Ki = 47.7 nM T32060 C2J0ZS 44335767 Ki = 44.6 nM T32060 C2TC7Y 44335888 Ki = 120.7 nM T32060 CPWJ26 44343212 Ki < 3162.28 nM T32060 C6N3XK 44345317 IC50 < 1000 nM T32060 CCU89V 44350664 Ki = 106 nM T32060 CUXH48 44352308 Ki = 1000 nM T32060 CJ80OW 44360984 Ki = 100 nM T32060 CS8K1A 44360992 Ki = 780 nM T32060 C3NZ7B 44361021 Ki = 310 nM T32060 C3LKN1 44364048 Ki = 10000 nM T32060 CX38YF 44364163 Ki = 10.2 nM T32060 C6M0VT 44364215 Ki = 30.9 nM T32060 C8DVZ6 44364514 Ki = 164 nM T32060 CMU02Q 44364616 Ki = 1.8 nM T32060 CJ0SZ2 44369910 Ki = 11.22 nM T32060 CZIP61 44369921 Ki = 691.83 nM T32060 CW2X3H 44369922 Ki = 977.24 nM T32060 CG5A2S 44369987 Ki = 7.244 nM T32060 CXIM47 44369992 Ki = 5.623 nM T32060 C1U9IX 44370125 Ki = 660.69 nM T32060 CM3W6Y 44370126 Ki = 891.25 nM T32060 C2SD5H 44370139 Ki = 2344.23 nM T32060 C9KI6O 44373282 Ki = 4000 nM T32060 CVL3U2 44374207 Ki = 480 nM T32060 CV8CP3 44374225 Ki = 1200 nM T32060 C04WKH 44374233 Ki = 270 nM T32060 CJ4A2U 44374299 Ki = 640 nM T32060 CVW0F4 44377901 Ki = 7.5 nM T32060 C2NE7B 44377927 Ki = 0.3 nM T32060 C1IDK8 44377928 Ki = 0.8 nM T32060 CD0T3J 44377939 Ki = 90 nM T32060 CN3FA5 44377954 Ki = 0.8 nM T32060 C49FLN 44377965 Ki = 51 nM T32060 CZK50H 44378001 Ki = 1.2 nM T32060 CVH02T 44378002 Ki = 3.7 nM T32060 C03SDF 44378003 Ki = 0.5 nM T32060 C62RSW 44378016 Ki = 0.8 nM T32060 C6Z9UH 44378022 Ki = 11.9 nM T32060 C7JB3Y 44378024 Ki = 1.6 nM T32060 C1UY7T 44378034 Ki = 1.5 nM T32060 C56ZJP 44378035 Ki = 6.6 nM T32060 CTC75H 44378076 Ki = 10.4 nM T32060 C3GTV5 44378077 Ki = 0.4 nM T32060 CS07QF 44378128 Ki = 2.7 nM T32060 CWU41H 44378141 Ki = 11 nM T32060 C9R5AX 44378333 Ki = 0.9 nM T32060 C6EMI4 44378348 Ki = 3.1 nM T32060 CJF5K0 44378369 Ki = 0.6 nM T32060 CJ3ZM8 44378381 Ki = 0.7 nM T32060 C2IA3N 44383324 Ki = 954 nM T32060 C25EZI 44383397 EC50 = 1100 nM T32060 C1XOB5 44387732 Ki = 0.3 nM T32060 CL54KN 44387733 Ki = 0.32 nM T32060 C80WKC 44387740 Ki = 2.4 nM T32060 CROA61 44387743 Ki = 1 nM T32060 C1M5OY 44387746 Ki = 0.68 nM T32060 CK36VZ 44387776 Ki = 2 nM T32060 CC0WK5 44387777 Ki = 0.66 nM T32060 CQ9WS8 44387780 Ki = 0.64 nM T32060 CQ85AW 44389003 Ki = 599 nM T32060 CB8L9M 44389309 Ki = 18.5 nM T32060 CI5P0E 44389321 Ki = 14.7 nM T32060 CVYR53 44389330 Ki = 17.9 nM T32060 C1B0VT 44389345 Ki = 9.67 nM T32060 C4MLR3 44389645 EC50 = 80 nM T32060 CUR07Z 44389646 EC50 = 30 nM T32060 C2VN8S 44392087 IC50 = 800 nM T32060 C6WAK2 44393173 Ki = 1548.82 nM T32060 COD15M 44394743 Ki = 460 nM T32060 C3RV6T 44395741 Ki = 109.6 nM T32060 C4B0OI 44397588 Ki = 398.11 nM T32060 C5FP0R 44397589 Ki = 794.33 nM T32060 CE3G8U 44397670 Ki = 794.33 nM T32060 CQR59X 44397731 Ki = 110 nM T32060 C8VJ5H 44397752 Ki = 102 nM T32060 C8EQU9 44397832 Ki = 7.5 nM T32060 CYDA14 44397846 Ki = 43 nM T32060 C0FUY7 44397929 Ki = 6.2 nM T32060 CX7O9S 44401041 Ki > 5454 nM T32060 C5XC2B 44401042 Ki = 22 nM T32060 CD56EA 44401105 Ki = 15 nM T32060 CW3PC2 44401106 Ki = 13 nM T32060 C9WH7P 44401164 Ki = 0.24 nM T32060 C9CWX1 44401194 Ki > 5454 nM T32060 CXT84G 44401243 Ki = 6 nM T32060 CR7H0V 44401244 Ki = 38 nM T32060 CFYR54 44402349 Ki = 255 nM T32060 CFH59G 44402373 Ki = 423 nM T32060 C6J2DO 44402413 Ki = 185 nM T32060 C8FK6D 44402415 Ki = 306 nM T32060 C9AJO5 44402449 Ki = 97 nM T32060 C9NJ8C 44402482 Ki = 189 nM T32060 C5RX3H 44402486 Ki = 5 nM T32060 C1X3WG 44402487 Ki = 65 nM T32060 CC30BR 44402509 Ki = 92 nM T32060 C8Y7SW 44402544 Ki = 307 nM T32060 C4EAG0 44402566 Ki = 95 nM T32060 CA56WF 44402586 Ki = 104 nM T32060 C4HEJ5 44402603 Ki = 11 nM T32060 C6K3RG 44402627 Ki = 306 nM T32060 C0SCV2 44402676 Ki = 36 nM T32060 C7YPE6 44402704 Ki = 3 nM T32060 CP6DL2 44402713 Ki = 193 nM T32060 CYH87E 44402816 Ki = 22 nM T32060 C1B4QL 44403095 Ki = 1008 nM T32060 C1YL7Z 44403098 Ki = 4451 nM T32060 CFV98A 44403101 Ki = 171 nM T32060 C6OY9S 44403102 Ki = 614 nM T32060 CH4SX6 44403105 Ki = 1335 nM T32060 C12FIH 44403106 Ki > 10000 nM T32060 C4LKC1 44404394 Ki = 5988 nM T32060 C3EJ4G 44404396 Ki > 10000 nM T32060 C0E9YL 44404412 Ki = 0.59 nM T32060 CR3Q7O 44404413 Ki = 0.44 nM T32060 CGCW03 44404417 Ki = 0.32 nM T32060 CFIS96 44404418 Ki = 0.31 nM T32060 C36EZX 44404422 Ki = 0.29 nM T32060 CW4E0R 44404423 Ki = 2.15 nM T32060 CM6JK9 44404428 Ki = 0.75 nM T32060 C1CFY7 44404437 Ki = 0.22 nM T32060 CPL38O 44404439 Ki = 0.17 nM T32060 CAH1M6 44404440 Ki = 1.06 nM T32060 CC7DU3 44404443 Ki = 0.17 nM T32060 CAS49R 44404446 Ki = 190 nM T32060 C4I7RN 44404449 Ki = 0.13 nM T32060 CN6TX1 44404450 Ki = 2.23 nM T32060 C4HWE2 44404453 Ki = 0.28 nM T32060 C5ZV3O 44404454 Ki = 0.05 nM T32060 C34KQU 44404456 Ki = 0.28 nM T32060 C4NX6R 44404457 Ki = 0.18 nM T32060 C7SZ6O 44404459 Ki = 0.28 nM T32060 C01GEA 44404460 Ki = 0.61 nM T32060 C92LED 44404463 Ki = 0.3 nM T32060 C20AJE 44404465 Ki = 1.24 nM T32060 C2L7DW 44404470 Ki = 1.07 nM T32060 CUVA58 44404608 Ki > 10000 nM T32060 C53KTE 44404616 Ki > 10000 nM T32060 C4XIR6 44404619 Ki > 10000 nM T32060 CW1BK6 44404623 Ki > 10000 nM T32060 CHG15M 44404887 Ki = 3000 nM T32060 CJ3ED5 44405445 Ki = 5600 nM T32060 CT5IP4 44405452 Ki = 22 nM T32060 C9YLW2 44405455 Ki = 16 nM T32060 C9Q7CS 44405466 Ki = 22 nM T32060 CCP9V7 44405469 Ki = 1100 nM T32060 C68OGK 44405489 Ki = 130 nM T32060 CX7ER9 44405490 Ki = 740 nM T32060 C3I8EC 44405492 Ki = 610 nM T32060 CYXC08 44405530 Ki = 140 nM T32060 CW20SO 44407327 EC50 > 1000 nM T32060 COY19S 44407335 Ki = 927 nM T32060 CW57QU 44407337 EC50 = 777 nM T32060 C6Z5PB 44407398 Ki = 181 nM T32060 C2Q5MJ 44407440 EC50 > 1000 nM T32060 CR1D5Y 44407453 EC50 = 638 nM T32060 CL94HP 44407460 Ki = 842 nM T32060 COH25L 44409031 Ki = 42 nM T32060 C4TZ7J 44409032 Ki = 54 nM T32060 C6I4CY 44409095 Ki = 511 nM T32060 CWX62Y 44409096 Ki = 136 nM T32060 CM6ZY0 44409097 Ki = 43 nM T32060 CJ8UB2 44409101 Ki = 565 nM T32060 C5K2ZG 44409124 Ki = 2547 nM T32060 CG87PW 44409290 Ki = 74 nM T32060 CI69ML 44409316 Ki = 53 nM T32060 CMP47G 44409317 Ki = 58 nM T32060 CIPR62 44409327 Ki = 65 nM T32060 CPDN92 44409332 Ki = 2385 nM T32060 CAO78Q 44411663 Ki = 2.1 nM T32060 C8NVH0 44411664 Ki = 3.9 nM T32060 C2Y8VK 44411667 Ki = 2.9 nM T32060 C38VWG 44411668 Ki = 4.4 nM T32060 C5Z2IY 44411674 Ki = 190 nM T32060 CU2EY5 44411847 Ki = 24 nM T32060 CD0OH1 44411864 Ki = 9.9 nM T32060 CTLN43 44411929 Ki = 22 nM T32060 CKX6D2 44411930 Ki = 6.1 nM T32060 CQ89KF 44411933 Ki = 52 nM T32060 CCJ1S9 44411934 Ki = 14 nM T32060 CL28ZA 44411935 Ki = 8.1 nM T32060 CG13DQ 44411936 Ki = 1.7 nM T32060 CQLM69 44412150 EC50 = 220 nM T32060 C0VIZ4 44412388 EC50 = 25 nM T32060 CZV87X 44412389 EC50 = 40 nM T32060 CA7CM1 44412403 EC50 = 416 nM T32060 C7R5WO 44412404 EC50 = 1120 nM T32060 CA1SO2 44412405 EC50 = 1080 nM T32060 C95IMP 44414051 Ki = 398.11 nM T32060 C9W3KV 44414057 Ki < 1258.93 nM T32060 C2JIS7 44414070 Ki = 501.19 nM T32060 CKM83W 44414105 Ki < 6309.57 nM T32060 C1MQU7 44414127 Ki < 794.33 nM T32060 C84CDF 44414132 Ki = 398.11 nM T32060 CX10RT 44414133 Ki = 398.11 nM T32060 C5HPJ4 44414150 Ki < 7943.28 nM T32060 C6ZTK1 44414164 Ki = 1000 nM T32060 CA4MG3 44414179 Ki = 630.96 nM T32060 CU7G6H 44414192 Ki < 1258.93 nM T32060 C5EO1B 44414209 Ki = 251.19 nM T32060 C9WJD2 44414217 Ki = 3162.28 nM T32060 CQ1H9S 44414233 Ki < 1258.93 nM T32060 CQ13GM 44414244 Ki < 1584.89 nM T32060 COY3V0 44414251 Ki = 158.49 nM T32060 CQ6K7F 44414267 Ki < 1258.93 nM T32060 CKG9P2 44414300 Ki < 10000 nM T32060 CU2FG6 44415569 Ki = 13.8 nM T32060 CDU6Y5 44415593 Ki = 1 nM T32060 CH0BY5 44415672 Ki = 1.2 nM T32060 CK59CO 44415689 Ki = 0.9 nM T32060 C7AZ5D 44415690 Ki = 2.2 nM T32060 CEVY54 44415704 Ki = 2.9 nM T32060 CS95TV 44416324 Ki = 170 nM T32060 CA5X0P 44416365 Ki = 200 nM T32060 CK9R1S 44420682 EC50 = 994 nM T32060 C6PBE9 44420683 Ki > 10000 nM T32060 C2TE3S 44425699 Ki = 5.012 nM T32060 CU52GB 44425701 Ki = 5.012 nM T32060 C9F1XP 44425702 Ki = 50.12 nM T32060 CR1QN5 44425703 Ki = 794.33 nM T32060 C5UZS7 44425704 Ki = 50.12 nM T32060 CN96FA 44425705 Ki = 1258.93 nM T32060 C1J9MY 44425706 Ki = 19.95 nM T32060 CPI52U 44425708 Ki = 5.012 nM T32060 C92AZG 44425714 Ki = 31.62 nM T32060 C7LP1B 44425717 Ki = 15.85 nM T32060 CX8TR0 44425719 Ki = 1.585 nM T32060 CJN6P4 44427818 Ki = 228 nM T32060 CW3F5H 44427820 Ki = 15.5 nM T32060 CYLO03 44427821 Ki = 92.7 nM T32060 CJY9L5 44427822 Ki = 46.9 nM T32060 CO46HS 44427823 Ki = 57.9 nM T32060 CFG0S3 44427824 Ki = 105 nM T32060 C7PK0M 44427825 Ki = 75.3 nM T32060 CDV6A3 44427826 Ki = 65.7 nM T32060 C65ZXC 44427827 Ki = 42.3 nM T32060 CZ0X7U 44427829 Ki = 545 nM T32060 C9U8YT 44427831 Ki = 695 nM T32060 C0C8AH 44427835 Ki = 88.7 nM T32060 C8EV3G 44427836 Ki = 15.4 nM T32060 CS9ND5 44427841 Ki = 47.1 nM T32060 COV6N3 44427842 Ki = 883 nM T32060 C7KBP0 44430566 Ki < 10000 nM T32060 CBP57S 44430955 Ki < 7943.28 nM T32060 CIZ54L 44430956 Ki < 1584.89 nM T32060 C1FHD3 44430958 Ki < 6309.57 nM T32060 CX0O2S 44430974 Ki < 3981.07 nM T32060 CQFV73 44430976 Ki < 1258.93 nM T32060 CG0CH7 44430979 Ki = 316.23 nM T32060 C14ZCW 44430984 Ki < 7943.28 nM T32060 CKZF16 44439165 Ki < 10000 nM T32060 CA4HZ3 44439167 Ki = 3162.28 nM T32060 CQ18PR 44439374 Ki = 9.6 nM T32060 CN9RH5 44439375 Ki = 5.4 nM T32060 C2X1FS 44439377 Ki = 150 nM T32060 CW2KQ1 44439378 Ki = 790 nM T32060 C2J9LG 44439379 Ki = 1.8 nM T32060 COKH57 44439380 Ki = 8.2 nM T32060 CO20GU 44439381 Ki = 9.9 nM T32060 C4KQ8C 44439384 Ki = 65 nM T32060 CQXS03 44439385 Ki = 4.6 nM T32060 C3OD9X 44441217 Ki = 42.66 nM T32060 CY29KE 44441218 Ki = 30.2 nM T32060 CRPB21 44441219 Ki = 17.38 nM T32060 C6JU0E 44441222 Ki = 40.74 nM T32060 CG4SU7 44441225 Ki = 17.38 nM T32060 C9E0FL 44447001 Ki = 0.09 nM T32060 CSJ4U5 44447002 Ki = 0.01 nM T32060 CL87PU 44447003 Ki = 0.45 nM T32060 CCD6B5 44447005 Ki = 0.3 nM T32060 CBH65G 44447007 Ki = 0.75 nM T32060 C8CF7X 44447008 Ki = 4.75 nM T32060 CN3EH7 44447010 Ki = 3 nM T32060 CYWP06 44447012 Ki = 0.1 nM T32060 C41KNM 44447013 Ki = 2.45 nM T32060 CE12BC 44447015 Ki = 0.95 nM T32060 CUD31L 44447018 Ki = 0.04 nM T32060 CNLX79 44447028 Ki = 0.95 nM T32060 CM8K1H 44447039 Ki = 0.55 nM T32060 C5IJW2 44447059 Ki = 0.08 nM T32060 CHXF10 44447061 Ki = 0.15 nM T32060 CG93OH 44447063 Ki = 0.25 nM T32060 C9KJR2 44447065 Ki = 0.5 nM T32060 C5QK8Z 44447067 Ki = 0.45 nM T32060 C7A6RP 44447068 Ki = 0.65 nM T32060 CM8P9A 44447070 Ki = 1.65 nM T32060 CK4HA6 44447072 Ki = 0.68 nM T32060 CZL95J 44451390 Ki = 90 nM T32060 CL14SE 44451393 Ki = 62 nM T32060 C32AJU 44451422 Ki = 130 nM T32060 CT5JO6 44451429 Ki = 51 nM T32060 C3Z7FI 44451927 IC50 > 10000 nM T32060 C57SBC 44451980 IC50 = 7900 nM T32060 CEST18 44451982 IC50 = 420 nM T32060 CRN4F8 44452007 IC50 = 2100 nM T32060 CG1C6X 44452142 IC50 = 620 nM T32060 CVAU93 44452222 IC50 = 1100 nM T32060 C0B3LC 44452327 IC50 = 1700 nM T32060 C63WNH 44452753 Ki = 8.7 nM T32060 CY9PG0 44452754 Ki = 0.78 nM T32060 CXCB32 44452783 Ki = 17 nM T32060 CD5J9B 44452784 Ki = 11 nM T32060 CI5R1U 44452785 Ki = 64 nM T32060 CX3PQ9 44452786 Ki = 47 nM T32060 C7E4KD 44452809 Ki = 9.1 nM T32060 CE7CQ0 44452810 Ki = 6.7 nM T32060 CNPZ39 44452831 Ki = 1200 nM T32060 CSM19Y 44452832 Ki = 11 nM T32060 CZE3G2 44453102 Ki = 38 nM T32060 C78NHG 44453103 Ki = 20 nM T32060 C5XTC7 44453127 Ki = 87 nM T32060 C6QHC2 44453128 Ki = 46 nM T32060 CQF0U6 44453129 Ki = 51 nM T32060 C4L6TY 44453652 Ki = 1200 nM T32060 CVN1O4 44453877 Ki = 50 nM T32060 C6BFI0 44456033 Ki = 257 nM T32060 C12XGE 44456400 Ki = 1318.26 nM T32060 C5RO6E 44461290 IC50 > 1000 nM T32060 CC9JB4 44461357 IC50 = 1.905 nM T32060 CI85BO 44461456 IC50 = 57.54 nM T32060 CE12QP 44461565 IC50 = 3.89 nM T32060 CQ2IX7 44461606 IC50 = 91.2 nM T32060 C5RM2Q 44461613 IC50 > 1000 nM T32060 CJ91XI 44461619 IC50 > 1000 nM T32060 CQX62Y 44461622 IC50 = 42.66 nM T32060 C80PVC 44461625 IC50 > 1000 nM T32060 CT09SU 44461626 IC50 > 1000 nM T32060 CR54MO 44461647 IC50 > 1000 nM T32060 C3XUF0 44461656 IC50 = 281.84 nM T32060 C5P3AW 44461799 IC50 > 1000 nM T32060 C52INO 44461800 IC50 = 141.25 nM T32060 C4DL5C 44469677 IC50 > 10000 nM T32060 CR74ZI 44473056 Ki = 33 nM T32060 C6PT2I 44473057 Ki = 46 nM T32060 C7CEY4 44473058 IC50 = 477 nM T32060 CRZK08 44473059 Ki = 619 nM T32060 CV3TN8 44473060 Ki = 854 nM T32060 C9OY3U 44517726 Ki = 630.96 nM T32060 CM23CO 44521013 Ki = 84 nM T32060 CT85QK 44538690 Ki = 0.89 nM T32060 CUQ0J7 44555369 EC50 > 1500 nM T32060 CY18IU 44555382 Ki = 0.15 nM T32060 C6WV2P 44559406 IC50 > 10000 nM T32060 CR8OX1 44562611 IC50 = 9.04 nM T32060 CL64BM 44562612 IC50 = 48.6 nM T32060 CVB0Q6 44562613 IC50 = 32.9 nM T32060 C02CWF 44562614 IC50 = 60.9 nM T32060 C7CSF8 44562615 IC50 = 48.9 nM T32060 CNJM41 44562616 IC50 = 58.1 nM T32060 C3VP6N 44562943 IC50 = 3.42 nM T32060 C7DS0M 44562944 IC50 = 34.7 nM T32060 C4XL2E 44562989 IC50 = 721 nM T32060 C4UG5R 44562990 IC50 = 2240 nM T32060 CY84FH 44563029 IC50 = 74.2 nM T32060 C5N9FG 44563030 IC50 = 1000 nM T32060 C5J6HU 44563054 IC50 = 651 nM T32060 C6B2FI 44563127 IC50 = 5570 nM T32060 CL0DS9 44563128 IC50 = 1550 nM T32060 C0J2GS 44563163 IC50 = 230 nM T32060 C67TOD 44563164 IC50 = 291 nM T32060 CL5HW8 44563165 IC50 = 172 nM T32060 C7BRD0 44563202 IC50 = 378 nM T32060 CDX3R8 44563203 IC50 = 88 nM T32060 C5QX2S 44563204 IC50 = 324 nM T32060 CF4ZK8 44563205 IC50 = 1.18 nM T32060 C3ZUH6 44563206 IC50 = 47.1 nM T32060 CJ9O6U 44563238 IC50 = 6.59 nM T32060 CB8P3I 44563239 IC50 = 3.54 nM T32060 CB9NG8 44563240 IC50 = 6.82 nM T32060 CN5U4V 44563241 IC50 = 51 nM T32060 CLJ7C2 44563242 IC50 = 429 nM T32060 C2OX9D 44563243 IC50 = 90.2 nM T32060 C1VQ5X 44563244 IC50 = 9.11 nM T32060 CLW0R9 44565334 Ki = 2790 nM T32060 C3KL2J 44565335 Ki = 1390 nM T32060 C96WDV 44565336 Ki = 737 nM T32060 C16EQJ 44565358 Ki = 6019 nM T32060 C12AGB 44565359 Ki = 954.99 nM T32060 CD86LA 44565360 Ki = 286 nM T32060 C5MU6R 44565361 Ki = 169.82 nM T32060 CS2ZF8 44565378 Ki = 9720 nM T32060 C58LTW 44565379 Ki = 522 nM T32060 C1S7DU 44565380 Ki = 3380 nM T32060 CZ7V1L 44565381 Ki = 575.44 nM T32060 CL5IP7 44565403 Ki = 181 nM T32060 CFL8O9 44565404 Ki = 102 nM T32060 C6BWZ9 44565405 Ki = 2089.3 nM T32060 CN6WE3 44565406 Ki = 1023.29 nM T32060 CMZ29A 44565418 Ki = 575 nM T32060 CG05ON 44565419 Ki = 426.58 nM T32060 C69TSL 44565420 Ki = 292 nM T32060 C2HQ7F 44565421 Ki = 676.08 nM T32060 CPRH81 44565433 Ki = 1819.7 nM T32060 C5I0KF 44565434 Ki = 371.54 nM T32060 C7T6QG 44565435 Ki = 1071.52 nM T32060 CW63CT 44565436 Ki = 376 nM T32060 CH39OA 44565454 Ki = 630.96 nM T32060 C2K9MN 44565455 Ki = 300 nM T32060 C0W7RH 44565456 Ki = 910 nM T32060 CWS6J1 44565457 Ki = 109.65 nM T32060 CVA67X 44568347 Ki = 3600 nM T32060 CGFE18 44572164 EC50 = 774 nM T32060 CWG32I 44572166 EC50 = 91 nM T32060 C9B3LM 44572168 EC50 = 349 nM T32060 CYS32A 44572170 EC50 = 51 nM T32060 CX93AL 44572172 EC50 = 235 nM T32060 C9PGC5 44572174 EC50 = 726 nM T32060 C07DQB 44572176 EC50 = 465 nM T32060 CS26GU 44572178 EC50 = 360 nM T32060 CJA7V6 44572180 EC50 = 2392 nM T32060 CYOJ47 44572207 EC50 = 330 nM T32060 C6GIR9 44572369 EC50 > 10000 nM T32060 C7WJS5 44572657 EC50 = 1396 nM T32060 C9QJB3 44572747 EC50 > 681 nM T32060 C6S2DJ 44572749 EC50 = 168 nM T32060 C97VKX 44572751 EC50 = 67 nM T32060 C2RV0K 44572755 EC50 = 1606 nM T32060 CQU5B9 44572759 EC50 = 2166 nM T32060 CYTA39 44572761 EC50 = 513 nM T32060 C6CGB5 44572798 EC50 = 437 nM T32060 C20GHO 44572800 EC50 = 1886 nM T32060 CJ1VI8 44572802 EC50 = 585 nM T32060 CLV5I8 44572804 EC50 = 1485 nM T32060 C43IDZ 44572806 EC50 = 613 nM T32060 CT64CF 44572808 EC50 = 247 nM T32060 CU25XD 44572810 EC50 = 508 nM T32060 CS7KZ5 44572812 EC50 = 4482 nM T32060 C6QFY7 44573002 EC50 > 1000 nM T32060 CP16NR 44573004 EC50 = 1929 nM T32060 CQ70OY 44573012 EC50 > 5000 nM T32060 CE95AX 44573014 EC50 = 547 nM T32060 CEC7J9 44573016 EC50 > 1000 nM T32060 CUB38Y 44573018 EC50 = 578 nM T32060 CPD63U 44574738 IC50 = 4600 nM T32060 CST84W 44579032 Ki > 10000 nM T32060 CV32GO 44579033 Ki > 10000 nM T32060 C61JVZ 44579034 Ki > 10000 nM T32060 CJ1WX8 44579464 Ki = 166 nM T32060 CNZ59J 44579538 Ki = 83 nM T32060 C5TKU6 44579715 Ki > 10000 nM T32060 C5NS6H 44581972 Ki = 60.26 nM T32060 CK8Z1P 44581973 Ki = 2.138 nM T32060 C3UQ9Z 44581974 Ki = 52.48 nM T32060 CA9XV2 44591684 Ki > 3200 nM T32060 C2OK6Y 44591772 Ki > 3100 nM T32060 CE0XV7 44591773 Ki = 323 nM T32060 CQL3J1 44591794 Ki > 3100 nM T32060 CX3T0N 44591796 Ki > 3100 nM T32060 CB0S4Z 44592109 IC50 = 165.96 nM T32060 CY75PU 44593425 Ki = 230 nM T32060 CQ12YR 44593444 IC50 = 144 nM T32060 C67KZG 44608359 IC50 = 10 nM T32060 CU3LE6 44626329 Ki = 130 nM T32060 CZHP95 44626357 EC50 = 41 nM T32060 C7NIU3 44628133 Ki = 251.19 nM T32060 CE6M8G 44628198 Ki > 10000 nM T32060 CERD02 44628200 Ki = 3162.28 nM T32060 CIM8C4 44628201 Ki = 31.62 nM T32060 C2EW5K 44628269 Ki = 794.33 nM T32060 CR4UX9 44629279 Ki = 79.43 nM T32060 C4AEZ5 44629280 Ki > 1000 nM T32060 CAGF30 44629348 Ki = 100 nM T32060 C1XQ8G 44629350 Ki > 10000 nM T32060 C0DLU3 45109862 IC50 = 300 nM T32060 C2J0GO 45278647 IC50 = 209 nM T32060 C7X3LG 45278648 IC50 = 46 nM T32060 CG64BP 45278720 IC50 = 92 nM T32060 CD9HF8 45278721 IC50 = 57 nM T32060 CYT87H 45278722 IC50 = 92 nM T32060 C8QK9C 45278723 IC50 = 75 nM T32060 C2M5HA 45278725 IC50 = 191 nM T32060 CXJ8L6 45278729 IC50 = 39 nM T32060 CAQ40Z 45278802 IC50 = 129 nM T32060 CARO27 45278803 IC50 = 441 nM T32060 CFG01K 45278804 IC50 = 133 nM T32060 CZ71RN 45278805 IC50 = 46 nM T32060 CFN4D9 45278806 IC50 = 376 nM T32060 CZN6M7 45278882 IC50 = 324 nM T32060 C6NT3Q 45278883 IC50 = 67.1 nM T32060 CA58GM 45278884 IC50 = 22.9 nM T32060 C21JKF 45278885 IC50 = 6.9 nM T32060 CS5BA4 45278886 IC50 = 4.1 nM T32060 C4TXE8 45278964 IC50 = 179 nM T32060 CPI26X 45278965 IC50 = 224 nM T32060 C1NR0P 45278966 IC50 = 354 nM T32060 CYK65H 45278967 IC50 = 1067 nM T32060 C0EGV6 45278968 IC50 = 1233 nM T32060 CWI2S0 45279043 IC50 = 4383 nM T32060 CN7V2L 45279044 IC50 = 245 nM T32060 C2AW3R 45279045 IC50 = 300 nM T32060 CF7O1A 45279046 IC50 = 333 nM T32060 CM46OZ 45279047 IC50 = 897 nM T32060 CB02TI 45279127 IC50 = 406 nM T32060 CS62HT 45279130 IC50 = 33 nM T32060 CRM38P 45279134 IC50 = 792 nM T32060 CEZ53Y 45279210 IC50 = 104 nM T32060 CPX18C 45279212 IC50 = 61 nM T32060 CJ0X2R 45279214 IC50 = 28 nM T32060 C3NW0C 45279216 IC50 = 39 nM T32060 CX73IH 45279218 IC50 = 40 nM T32060 CGNC19 45279298 IC50 = 408 nM T32060 C8CPD7 45279300 IC50 = 10 nM T32060 CP4GI2 45279384 IC50 = 92 nM T32060 CX2ND5 45279386 IC50 = 105 nM T32060 CX5ST2 45279664 IC50 = 213 nM T32060 CKQ7S3 45279666 IC50 = 232 nM T32060 C91IRB 45279668 IC50 = 151 nM T32060 C12WRL 45279755 IC50 = 153 nM T32060 C3SUQ1 45279757 IC50 = 192 nM T32060 C63LSI 45279759 IC50 = 333 nM T32060 C0CHF4 45482789 IC50 = 750 nM T32060 CQ9FN0 45483190 Ki = 125.89 nM T32060 CEZW26 45483246 Ki = 309.03 nM T32060 CLO70J 45483261 Ki = 23.44 nM T32060 C2BW1S 45483262 Ki = 102.33 nM T32060 C7LD5K 45483269 Ki = 4.571 nM T32060 CG5TR7 45483288 Ki = 6.457 nM T32060 CHOK19 45483329 Ki = 630.96 nM T32060 C9NK6I 45485725 EC50 = 65 nM T32060 CVK8W9 45485742 EC50 = 308 nM T32060 CD80KX 45485751 EC50 = 254 nM T32060 CNX23T 45485779 EC50 = 114 nM T32060 CO6Z1P 45485781 EC50 = 1090 nM T32060 C9CV1H 45486652 Ki = 3.3 nM T32060 CY8T1Z 45486653 Ki = 0.22 nM T32060 C1WBI2 45486654 Ki = 2.5 nM T32060 C3ME0C 45486656 Ki = 0.61 nM T32060 C2AK3J 45486657 Ki = 0.54 nM T32060 C0VF7N 45486658 Ki = 0.82 nM T32060 CLOH56 45486664 Ki = 0.33 nM T32060 C5IV3W 45486665 Ki = 0.25 nM T32060 C0I6YB 45486671 Ki = 0.36 nM T32060 C12ELO 45486672 Ki = 0.99 nM T32060 C54GSK 45486673 Ki = 17.6 nM T32060 CD28FO 45486677 Ki = 0.19 nM T32060 C2GLK8 45486678 Ki = 2.1 nM T32060 CL6H8C 45486679 Ki = 0.96 nM T32060 C2TL5C 45486680 Ki = 1.9 nM T32060 CXQ5Z0 45486688 Ki = 0.26 nM T32060 CGZ62R 45486694 Ki = 0.15 nM T32060 C3W8EK 45486695 Ki = 0.43 nM T32060 C40DYQ 45486696 Ki = 0.34 nM T32060 CFLI93 45486697 Ki = 14.3 nM T32060 CBEF38 45486702 Ki = 0.66 nM T32060 CEF0H7 45486708 Ki = 0.55 nM T32060 CH9LW6 45486710 Ki = 0.42 nM T32060 C3LEN4 45486711 Ki = 3.2 nM T32060 C7NO8W 45486713 Ki = 0.84 nM T32060 CI4PE6 45486714 Ki = 0.43 nM T32060 CXI5R2 45486715 Ki = 0.41 nM T32060 CLID23 45486716 Ki = 0.12 nM T32060 CFB39Y 45486717 Ki = 0.69 nM T32060 CT51UF 45486721 Ki = 0.63 nM T32060 CIF10P 45486722 Ki = 4 nM T32060 CUZ79F 45486723 Ki = 0.58 nM T32060 CA39DM 45486724 Ki = 0.99 nM T32060 C9X2NP 45486725 Ki = 0.84 nM T32060 C3LX5I 45486726 Ki = 2.1 nM T32060 CTC15H 45486727 Ki = 0.91 nM T32060 CR25SJ 45486729 Ki = 16.2 nM T32060 CES7G9 45486731 Ki = 1.4 nM T32060 CX74NQ 45486732 Ki = 0.86 nM T32060 C4RTL1 45486733 Ki = 0.31 nM T32060 CM08SQ 45486737 Ki = 1.4 nM T32060 CFEK40 45486738 Ki = 0.28 nM T32060 CQMJ83 45486820 Ki = 1800 nM T32060 CJN7X0 45486824 Ki = 2 nM T32060 C9BSL5 45486891 Ki = 6 nM T32060 CXT96Y 45815848 Ki > 10000 nM T32060 CV7C2M 45827434 Ki = 5434 nM T32060 CIV92F 46214153 Ki = 42 nM T32060 C16KNO 46216770 Ki = 400 nM T32060 CRT07W 46216771 Ki = 223 nM T32060 C7M9XU 46216789 Ki = 365 nM T32060 C5FQ4S 46224879 Ki = 1 nM T32060 CF6BQ7 46228422 EC50 = 1311 nM T32060 C23DJK 46228430 EC50 = 578 nM T32060 CTES15 46228437 EC50 = 70 nM T32060 CZ5MW9 46228438 EC50 = 236 nM T32060 C98NCA 46230046 Ki = 1980 nM T32060 C3LMQ6 46230047 EC50 > 705 nM T32060 C0D4IZ 46230048 EC50 > 10000 nM T32060 C6UMX7 46230049 Ki = 334 nM T32060 C87JZL 46230094 Ki = 397 nM T32060 CINK61 46230095 Ki = 184 nM T32060 C6N7AF 46230096 Ki > 10000 nM T32060 C7WO5P 46230097 EC50 = 248 nM T32060 CP0T5Y 46230098 EC50 = 70 nM T32060 CPA62G 46230099 EC50 = 130 nM T32060 CWQD49 46230100 Ki = 364 nM T32060 CTE69Y 46230651 Ki = 21 nM T32060 CXUL12 46232559 IC50 = 2.6 nM T32060 CU2RG8 46232560 IC50 = 7.1 nM T32060 C9RQ8U 46232586 IC50 = 13.2 nM T32060 C2B3ZP 46232587 IC50 = 4.2 nM T32060 C3I8TO 46232588 IC50 = 9.4 nM T32060 COW9V6 46232589 IC50 = 16.3 nM T32060 CGV2J5 46232620 IC50 = 19.5 nM T32060 CWHG97 46232621 IC50 = 3.4 nM T32060 CUQW08 46232622 IC50 = 0.7 nM T32060 C5REP7 46232623 IC50 = 11.6 nM T32060 C2QOW0 46232652 IC50 = 13.1 nM T32060 C9I7XS 46232653 IC50 = 0.5 nM T32060 C5D0BH 46232654 IC50 = 34.6 nM T32060 C5PAL9 46232689 IC50 = 59.9 nM T32060 CT5C0M 46232690 IC50 = 29.1 nM T32060 CF53BL 46232691 IC50 = 5.1 nM T32060 CE1ID7 46232729 IC50 = 7.7 nM T32060 CN0CO9 46232730 IC50 = 171 nM T32060 C0VXA5 46232731 IC50 = 70.8 nM T32060 C1C4OF 46232732 IC50 = 142 nM T32060 CMR8O9 46232770 IC50 = 180 nM T32060 CTY9H7 46232771 IC50 = 136 nM T32060 C5TBE8 46232772 IC50 = 2210 nM T32060 COH03R 46232773 IC50 = 726 nM T32060 CZ2W7X 46232817 IC50 = 72.5 nM T32060 C0N4YP 46232818 IC50 = 35.9 nM T32060 CTJ89I 46232819 IC50 = 85.8 nM T32060 CS98DM 46232820 IC50 = 221 nM T32060 C8P3HD 46232858 IC50 = 51 nM T32060 CP04TS 46232859 IC50 = 292 nM T32060 C8W0IJ 46232860 IC50 = 561 nM T32060 CF5M2T 46232861 IC50 = 75 nM T32060 C21CHG 46232975 IC50 = 8.3 nM T32060 CO41KX 46232976 IC50 = 12.7 nM T32060 CIK94R 46232977 IC50 = 664 nM T32060 CB67ST 46232978 IC50 = 180 nM T32060 CRU0F7 46233014 IC50 = 6.2 nM T32060 C3GO2H 46233391 EC50 = 120 nM T32060 C42SVX 46700866 IC50 > 10000 nM T32060 CD0K6E 46700867 IC50 = 6800 nM T32060 C6K0MF 46830177 Ki = 12.8 nM T32060 C5TC2S 46830335 IC50 > 10000 nM T32060 C1K7FL 46830336 IC50 > 10000 nM T32060 C7G3AC 46833072 Ki = 12 nM T32060 CICY27 46833073 Ki = 8.6 nM T32060 CBO0R4 46833074 Ki = 0.6 nM T32060 C6G1DY 46833075 Ki = 0.7 nM T32060 CW6O7R 46833076 Ki = 4.1 nM T32060 CI4DB9 46833077 Ki = 287 nM T32060 CWU46E 46833370 Ki = 5.3 nM T32060 CZY08H 46833371 Ki = 4.3 nM T32060 CRCS34 46833372 Ki = 2.2 nM T32060 C5L9IJ 46833373 Ki = 5.1 nM T32060 CXIE19 46833374 Ki = 28 nM T32060 C8WCT0 46833678 Ki = 2.2 nM T32060 C1N4KX 46842383 IC50 > 10000 nM T32060 CC62SX 46866711 IC50 = 122 nM T32060 CHIW05 46880277 IC50 = 175 nM T32060 CK8A1O 46880462 Ki > 10000 nM T32060 C9KDP4 46880463 Ki > 10000 nM T32060 CODR73 46880498 Ki > 10000 nM T32060 CHJ5Y6 46880566 Ki > 10000 nM T32060 CE9PG2 46880567 Ki > 10000 nM T32060 C01PGO 46880568 Ki > 10000 nM T32060 CS7L4X 46880569 Ki > 10000 nM T32060 C0PXY7 46880628 Ki > 10000 nM T32060 CD37LU 46880629 Ki > 10000 nM T32060 CUY89F 46880630 Ki > 10000 nM T32060 C4P6XS 46880631 Ki > 10000 nM T32060 CJ53KF 46880672 Ki > 10000 nM T32060 CYJC08 46880673 Ki > 10000 nM T32060 C1RI9O 46880674 Ki > 10000 nM T32060 C2MC4K 46881463 Ki = 1584.89 nM T32060 CSQ4C9 46881468 Ki = 2511.89 nM T32060 C5BFY9 46884102 Ki = 13.7 nM T32060 C1ORQ0 46884137 EC50 = 153 nM T32060 C3BW2P 46884138 EC50 = 500 nM T32060 CB8GE1 46884818 IC50 > 10000 nM T32060 C4MQ0A 46884856 IC50 > 10000 nM T32060 CCNT25 46884898 IC50 > 10000 nM T32060 C3MSG2 46885027 IC50 > 10000 nM T32060 CB7XI0 46885213 IC50 > 10000 nM T32060 C3MPJ7 46890808 Ki = 2.1 nM T32060 C60OHX 46901596 Ki = 155 nM T32060 C4VIO7 46901598 Ki = 88 nM T32060 CT5S4Q 46901603 Ki > 10000 nM T32060 C7KO6F 46901762 Ki > 10000 nM T32060 CYQ3L9 46901908 Ki = 28 nM T32060 CX3AE0 46901909 Ki = 11 nM T32060 C2ULG1 46927928 IC50 = 152 nM T32060 CK21VU 46927929 IC50 = 233 nM T32060 CG7WR2 46933089 Ki = 79.43 nM T32060 CW4N5K 46933090 Ki = 63.1 nM T32060 CZO5F8 46933091 Ki = 50.12 nM T32060 CX7R3H 46933845 Ki > 10000 nM T32060 CUTX67 46934428 IC50 = 118 nM T32060 CV8A5L 46937339 EC50 = 894 nM T32060 C6J4TV 46946859 Ki = 4.95 nM T32060 C3XFG4 47029237 Ki > 10000 nM T32060 C2LZJ0 49783209 Ki = 1776 nM T32060 C57SMG 49783415 Ki > 10000 nM T32060 C0TG6I 49783419 Ki > 10000 nM T32060 CD53RT 49833882 Ki = 501.19 nM T32060 C5Y4DE 49833883 Ki = 398.11 nM T32060 CGT73Y 49833884 Ki = 125.89 nM T32060 CKL16R 49833886 Ki = 251.19 nM T32060 C3KSZ8 49834050 Ki = 316.23 nM T32060 C9QS2K 49834051 Ki > 794.33 nM T32060 CF4SX0 49834052 Ki = 199.53 nM T32060 C52GPW 49834053 Ki = 100 nM T32060 CO20JE 49836187 Ki = 1995.26 nM T32060 CG0LF8 49836189 Ki = 3981.07 nM T32060 C0UI3V 49836294 Ki = 398.11 nM T32060 CT7CV0 49836295 Ki = 125.89 nM T32060 CVG9X5 49836296 Ki > 758.58 nM T32060 C5E2ZK 49836298 Ki = 79.43 nM T32060 CYJW87 49836299 Ki = 79.43 nM T32060 C0MS8L 49836300 Ki = 39.81 nM T32060 CR40BA 49836386 IC50 = 840 nM T32060 CKS86Q 49836409 Ki = 100 nM T32060 C8E6WA 49836410 Ki = 50.12 nM T32060 CE0PN6 49836411 Ki = 630.96 nM T32060 C0I4EC 49836412 Ki = 63.1 nM T32060 C5HU1D 49836413 Ki = 79.43 nM T32060 C1UGC7 49836414 Ki = 100 nM T32060 C0M5XC 49836496 IC50 = 28000 nM T32060 C5ZV2Y 49836522 Ki = 316.23 nM T32060 C1JTH9 49836524 Ki = 19.95 nM T32060 C90XTY 49836525 Ki = 12.59 nM T32060 CK5QW9 49836526 Ki = 19.95 nM T32060 C8RL7C 49836527 Ki = 630.96 nM T32060 CNM9X8 49836528 Ki = 31.62 nM T32060 COK75S 49836633 Ki = 15.85 nM T32060 CZ6F7L 49836634 Ki = 50.12 nM T32060 CRM28S 49836635 Ki = 50.12 nM T32060 CA6QB8 49836636 Ki = 398.11 nM T32060 CB81YG 49836637 Ki = 25.12 nM T32060 CX43UC 49836639 Ki = 316.23 nM T32060 CEBP01 49836737 Ki = 398.11 nM T32060 CCMJ40 49836738 Ki = 100 nM T32060 CY1UR9 49836739 Ki > 1995.26 nM T32060 C3OK9Y 49836740 Ki = 398.11 nM T32060 C26NFU 49836741 Ki = 125.89 nM T32060 C6YM8W 49836842 Ki > 1995.26 nM T32060 C4R2YS 49850567 Ki = 158.49 nM T32060 C07JTU 49850570 Ki = 316.23 nM T32060 CK68QR 49850672 Ki = 199.53 nM T32060 CN5XR1 49850772 Ki = 398.11 nM T32060 CR4EZ0 49850870 Ki = 794.33 nM T32060 C5K4EC 49850872 Ki = 251.19 nM T32060 C8AW0R 49850874 Ki = 79.43 nM T32060 C6OQV2 49862237 Ki > 1000 nM T32060 C6IW4Q 49862238 Ki > 1000 nM T32060 CIA24C 49863566 IC50 = 107 nM T32060 CZB85K 49863567 IC50 = 163 nM T32060 C7V6WO 49863654 IC50 = 213 nM T32060 CH36GC 49863692 IC50 = 221 nM T32060 C39VLG 49863693 IC50 = 666 nM T32060 CKF87D 49863694 IC50 = 22 nM T32060 CZF5Q2 49863695 IC50 = 352 nM T32060 CFTZ59 49863717 IC50 = 832 nM T32060 C7IK0Y 49863741 IC50 = 54 nM T32060 C1GR9V 49863742 IC50 = 221 nM T32060 CRQ7U4 49863743 IC50 = 953 nM T32060 CF2TO6 49863774 IC50 = 153 nM T32060 C7Y8OQ 49863775 IC50 = 874 nM T32060 C24EAI 49863776 IC50 = 135 nM T32060 CM72WN 49863778 IC50 = 410 nM T32060 CZR6T8 49863794 IC50 = 210 nM T32060 CB13XF 49863795 IC50 = 17 nM T32060 C6GB5R 49863847 IC50 = 37 nM T32060 C8PQB0 49863849 IC50 = 33 nM T32060 C1EKY3 49863851 IC50 = 25 nM T32060 CS80EL 49863853 IC50 = 39 nM T32060 C4HB5K 49863957 IC50 = 34 nM T32060 C18ICN 49863958 IC50 = 36 nM T32060 C8H6GV 49863959 IC50 = 386 nM T32060 CMRQ30 49863961 IC50 = 50 nM T32060 C9KIU1 49864289 IC50 = 88 nM T32060 CHO9C0 49864292 IC50 = 50 nM T32060 C90MTG 49864602 IC50 = 172 nM T32060 C5BCS4 49864722 IC50 = 1423 nM T32060 CKZO79 49864723 IC50 = 389 nM T32060 C74LZS 49864724 IC50 = 218 nM T32060 CZ2SA8 49864841 Ki = 7.943 nM T32060 C2OCZ3 49864885 Ki > 5011.87 nM T32060 CS4Z8A 49864886 Ki = 39.81 nM T32060 CN8XT2 49865829 Ki > 10000 nM T32060 C1FMH5 49865830 Ki > 10000 nM T32060 C1CX5F 49865831 Ki > 10000 nM T32060 C8RYW1 49865832 Ki > 10000 nM T32060 C5ED3T 49865833 Ki > 10000 nM T32060 CAU15V 49865885 Ki > 10000 nM T32060 CLS0F3 49865886 Ki > 10000 nM T32060 CIG69Z 49865887 Ki > 10000 nM T32060 C5YEG8 49865888 Ki > 10000 nM T32060 CXP91V 49865889 Ki > 10000 nM T32060 C98TVK 49865890 Ki > 10000 nM T32060 C2RY0J 50878551 EC50 = 2.8 nM T32060 C1W6TV 50898777 Ki = 6309.57 nM T32060 CXMZ73 50898778 Ki > 10000 nM T32060 CYGD56 50899654 IC50 = 166 nM T32060 CBLK68 50899745 IC50 = 113 nM T32060 CJI9U2 50899747 IC50 = 55 nM T32060 CU7TK4 50899749 IC50 = 47 nM T32060 CW9SV5 50942111 EC50 = 2634 nM T32060 CX48AD 51002362 Ki = 2374 nM T32060 C8TA1J 51003550 IC50 = 1462 nM T32060 CQ1UJ7 51003551 IC50 = 48 nM T32060 CGMI37 51003586 IC50 = 455 nM T32060 CE4KP1 51050257 Ki > 10000 nM T32060 CI90RZ 51094588 EC50 > 10000 nM T32060 CIJT81 51111982 Ki = 59 nM T32060 C2HGK8 51122451 Ki = 392 nM T32060 CIWA18 52938727 Ki = 245 nM T32060 C6XY8V 52938728 Ki = 174 nM T32060 CX5ZB8 52940714 IC50 = 842 nM T32060 C9C0NB 52940734 Ki = 14 nM T32060 C0UXM7 52941358 Ki = 0.568 nM T32060 CTM81E 52941423 Ki = 3.85 nM T32060 CM4XO6 52941718 Ki > 1000 nM T32060 CE26GV 52941856 IC50 = 458 nM T32060 CH86KJ 52941866 IC50 = 256 nM T32060 CE6R7D 52942615 Ki = 9.43 nM T32060 CX2E5H 52942854 Ki = 9.53 nM T32060 CU8WA5 52942916 Ki = 11.4 nM T32060 C7OZN4 52944115 Ki = 12.59 nM T32060 CZ21PJ 52944292 IC50 = 263 nM T32060 CBU2Z6 52944379 Ki = 55.9 nM T32060 C59ASG 52945060 Ki = 16.1 nM T32060 C2TK7W 52945494 IC50 = 490 nM T32060 CPD0Y9 52945500 IC50 = 54 nM T32060 CL7OG0 52945537 IC50 = 274 nM T32060 CHFI03 52945539 IC50 = 69 nM T32060 C4SH8M 52945840 Ki = 29.5 nM T32060 CNQF49 52945978 Ki = 158.49 nM T32060 CRIV53 52946792 Ki = 12.5 nM T32060 C4S8JC 52946835 Ki = 36.8 nM T32060 CS3OD1 52947342 Ki = 3.55 nM T32060 CCOQ59 52947343 Ki = 1.13 nM T32060 C6YB2T 52947380 Ki = 34.4 nM T32060 CRH1P6 52947969 IC50 = 35 nM T32060 CD17LV 52948101 Ki = 65.7 nM T32060 C7IR4Q 52948256 Ki = 52 nM T32060 CJ6OP5 52948620 Ki = 25.3 nM T32060 CFN80U 52949206 IC50 = 744 nM T32060 CLOB90 52949351 Ki = 55 nM T32060 C0RUM1 52949810 Ki = 24.7 nM T32060 CS6O4B 52949885 Ki = 1.26 nM T32060 CILY85 52950060 Ki = 2.06 nM T32060 CPVM58 52950169 Ki = 8.84 nM T32060 CPA2G4 52951481 Ki = 6280 nM T32060 CYP0I3 52951482 Ki = 1130 nM T32060 C4IV2J 53248158 Ki = 2060 nM T32060 C03JEZ 53248159 Ki = 98 nM T32060 C2G0ZY 53248208 Ki = 4800 nM T32060 C2UKM3 53248209 Ki > 8800 nM T32060 C8KW9J 53248210 Ki = 3000 nM T32060 C87SLP 53248211 Ki = 274 nM T32060 CVD7E5 53248212 Ki = 3240 nM T32060 CX6KG9 53248213 Ki = 212 nM T32060 C63MQD 53248256 Ki > 10000 nM T32060 CG2O7F 53248257 Ki = 4800 nM T32060 CRK87G 53248258 Ki = 3030 nM T32060 C73WQX 53248259 Ki = 3290 nM T32060 CKOV84 53248260 Ki = 3540 nM T32060 C09IXA 53248261 Ki = 272 nM T32060 C5K7NT 53248298 Ki = 1910 nM T32060 CN4SY6 53248395 Ki = 2580 nM T32060 C0AY5O 53317923 EC50 = 40 nM T32060 CC0T6E 53317924 EC50 = 2046 nM T32060 C1T3AI 53317925 EC50 = 762 nM T32060 C61DNP 53320009 IC50 = 366 nM T32060 C9ZDR5 53320010 IC50 = 760 nM T32060 C40VGZ 53321865 EC50 = 5165 nM T32060 C7LE3I 53321947 EC50 = 2310 nM T32060 CC3DB8 53321948 EC50 = 32 nM T32060 CQLK01 53322638 IC50 = 704 nM T32060 CUNP37 53323196 EC50 = 63 nM T32060 C32YWL 53324045 Ki = 1000 nM T32060 CJ9I7U 53324165 EC50 = 138 nM T32060 CQVR02 53324327 EC50 = 1227 nM T32060 CR4W9L 53324553 Ki = 6022 nM T32060 CN8X4Z 53324629 EC50 = 585 nM T32060 C8DL1N 53324630 EC50 = 648 nM T32060 C35GJZ 53325137 Ki = 100000 nM T32060 CRQF15 53325242 Ki = 1000 nM T32060 CB37XF 53325861 Ki > 10000 nM T32060 C2ZFP8 53325935 EC50 = 2348 nM T32060 CNE6Q8 53325936 EC50 = 7774 nM T32060 C8VUJ6 53325937 EC50 = 3 nM T32060 CMB09H 53325938 EC50 = 2676 nM T32060 CU7W2I 53362841 Ki = 2000 nM T32060 CMOZ61 53475319 Ki = 2841 nM T32060 CWH50X 53499206 Ki > 10000 nM T32060 C7HP2L 53524618 Ki > 10000 nM T32060 C9PQ6Y 53550713 Ki > 10000 nM T32060 CR07QE 54186017 Ki = 3.3 nM T32060 CY18NZ 54189746 IC50 = 1019 nM T32060 C48CEL 54576149 IC50 = 174.9 nM T32060 C6PDR1 54576153 IC50 = 126 nM T32060 CX4OJ6 54576369 IC50 = 185 nM T32060 CA0O2M 54576371 IC50 = 204.5 nM T32060 CY67DI 54576594 IC50 = 579 nM T32060 CWUK35 54576597 IC50 = 78.3 nM T32060 C40IGO 54576800 IC50 = 91 nM T32060 CP4CV6 54576803 IC50 = 327 nM T32060 C4H3DT 54576804 IC50 = 71 nM T32060 CG24OE 54577010 IC50 = 75 nM T32060 CYZX34 54577012 IC50 = 105 nM T32060 C2WQE9 54577014 IC50 = 133 nM T32060 C83FGA 54577018 IC50 = 216.8 nM T32060 CWA58G 54577234 IC50 = 29.4 nM T32060 CA83GC 54577236 IC50 = 13.2 nM T32060 CJA0P6 54577243 IC50 = 231.5 nM T32060 C0NBJ7 54577435 IC50 = 144 nM T32060 CYW50O 54577439 IC50 = 253 nM T32060 C8YAZ5 54577443 IC50 = 62.7 nM T32060 C3P0LZ 54577446 IC50 = 294 nM T32060 CA94CQ 54577447 IC50 = 72.5 nM T32060 CE64WZ 54577448 IC50 = 646 nM T32060 CJS4H9 54577449 IC50 = 270 nM T32060 CMR6C3 54577665 IC50 = 70.8 nM T32060 CS9G8L 54577668 IC50 = 24 nM T32060 CA8J7E 54577670 IC50 = 244 nM T32060 C3P2KF 54577879 IC50 = 19 nM T32060 C9GFP0 54577882 IC50 = 64.8 nM T32060 C6KY9M 54577886 IC50 = 117.9 nM T32060 CES29I 54578098 IC50 = 31 nM T32060 CQ67LT 54578099 IC50 = 141 nM T32060 CAPC31 54578102 IC50 = 27.8 nM T32060 C12XBJ 54578547 IC50 = 32 nM T32060 CP24ZC 54579002 IC50 = 40.6 nM T32060 CXQK40 54579004 IC50 = 241 nM T32060 CZC81X 54579005 IC50 = 19 nM T32060 CSW18T 54579229 IC50 = 247.6 nM T32060 C5HC0P 54579233 IC50 = 58.6 nM T32060 CA4E9U 54579450 IC50 = 839.9 nM T32060 C3L1IB 54579451 IC50 = 1011 nM T32060 CTQ08M 54586179 Ki = 1.4 nM T32060 C0J8XZ 54598062 Ki = 192 nM T32060 CL5I1R 54753271 Ki = 1270 nM T32060 C28MPB 55253945 EC50 > 10000 nM T32060 CC57DS 55254237 EC50 = 5620 nM T32060 CW89BT 56595402 Ki > 1000 nM T32060 C4C3XQ 56595529 Ki > 1000 nM T32060 CA54LD 56597090 Ki = 0.6 nM T32060 CK9SG4 56781741 Ki = 3654 nM T32060 CY2S8M 56820088 Ki = 3324 nM T32060 CUMB38 56834972 IC50 = 77 nM T32060 C1ZG7A 56933434 Ki = 3.7 nM T32060 CO0N2W 56943599 Ki = 7.7 nM T32060 C3DF5Z 56943600 Ki = 0.6 nM T32060 C19BDH 56943695 Ki = 2.3 nM T32060 CS7K3T 56943891 Ki = 12 nM T32060 CZ4L3S 56944082 Ki = 17 nM T32060 C5NI3K 56944086 Ki = 2700 nM T32060 C37BYO 56944186 Ki = 11 nM T32060 C9UOZ6 56944189 Ki = 13 nM T32060 CH7V9J 56944190 Ki = 4.9 nM T32060 CE49MC 56944191 Ki = 9 nM T32060 CX2RP5 56944287 Ki = 3.6 nM T32060 CB0P9N 56944383 Ki = 0.5 nM T32060 CEQ7I3 56944384 Ki = 0.8 nM T32060 CHWI01 56944473 Ki = 8.5 nM T32060 C6Y4ZQ 56944564 Ki = 1.5 nM T32060 C3B0MZ 56944565 Ki = 0.4 nM T32060 CI4KW0 56944664 Ki = 26 nM T32060 C39YHD 56944665 Ki = 0.6 nM T32060 C1W3GL 56944666 Ki = 1.7 nM T32060 C7J4UT 56944667 Ki = 2.1 nM T32060 CZT80U 56944668 Ki = 2.8 nM T32060 CTW2F5 56944763 Ki = 1.8 nM T32060 C50WEX 56944764 Ki = 3.5 nM T32060 CX0ZW2 56944859 Ki = 0.7 nM T32060 CF9V3Q 56945045 Ki = 8.1 nM T32060 CE4S5M 56945046 Ki = 13 nM T32060 CHN2F6 56949640 Ki = 6405 nM T32060 C1TC7Q 56963799 Ki = 1355 nM T32060 CUL4N1 56964693 Ki = 131 nM T32060 CQ5TP0 56964794 Ki = 180 nM T32060 CDGZ96 57326583 Ki = 1106 nM T32060 C20ILW 57326584 Ki = 92 nM T32060 CD9I4N 57334553 IC50 = 39.2 nM T32060 C6H9UV 57345617 Ki = 317 nM T32060 CZU6L2 57345618 Ki = 566.6 nM T32060 CK9G8H 57345619 Ki = 510.3 nM T32060 CATM39 57390694 Ki = 696 nM T32060 C6S0IE 57390695 Ki = 1003 nM T32060 CV08WY 57391216 Ki = 27 nM T32060 CD75YK 57391306 Ki = 222 nM T32060 C07PMA 57391307 Ki = 60 nM T32060 COA60R 57391358 Ki = 0.8 nM T32060 C7UC1O 57391359 Ki = 3.5 nM T32060 CNLK91 57391360 Ki = 1.5 nM T32060 CV7N9Z 57391692 IC50 = 1683 nM T32060 CQO80V 57391693 IC50 = 3450 nM T32060 CWT20M 57393083 Ki = 41 nM T32060 CTX71S 57393122 Ki = 5.6 nM T32060 CTF5M7 57393393 IC50 > 10000 nM T32060 C9QT8H 57393432 IC50 = 452 nM T32060 CADH19 57394285 Ki = 163 nM T32060 C0WA3H 57394810 Ki = 112 nM T32060 CKL2B3 57394858 Ki = 5.7 nM T32060 CNGJ92 57394859 Ki = 0.6 nM T32060 CM7FS9 57394860 Ki = 1.7 nM T32060 CVZ5Q2 57395160 IC50 = 986 nM T32060 CD4A3P 57396484 Ki = 23 nM T32060 C4EXS6 57396571 Ki = 19.8 nM T32060 CY4JR5 57396622 Ki = 1.4 nM T32060 C6HBG0 57396813 Ki = 3700 nM T32060 C80SUY 57396884 IC50 = 5980 nM T32060 C5FU4X 57396934 IC50 > 10000 nM T32060 C3GW6L 57398351 Ki = 121 nM T32060 CO50ZB 57398352 Ki = 1129 nM T32060 CQ0D5K 57398388 Ki = 1.8 nM T32060 CNZ6E8 57398389 Ki = 18 nM T32060 CM8S6E 57398674 IC50 = 281 nM T32060 CBXQ64 57398675 IC50 = 1550 nM T32060 CJ41PW 57399432 Ki = 159 nM T32060 CO3B4P 57399494 Ki = 411.5 nM T32060 C0R6QM 57400053 Ki = 0.4 nM T32060 CN7G6D 57400054 Ki = 2.6 nM T32060 CO98FL 57400055 Ki = 1.9 nM T32060 CUQZ68 57400351 IC50 = 1859 nM T32060 CZX05B 57401706 Ki = 26 nM T32060 CYN38R 57401819 Ki = 81 nM T32060 CO0XD2 57401820 Ki = 53 nM T32060 CHG0A7 57401861 Ki = 5.9 nM T32060 CA51WJ 57401862 Ki = 4.3 nM T32060 C3SB2U 57401863 Ki = 2.8 nM T32060 C92HON 57402951 Ki = 1038 nM T32060 CX0B5M 57403525 Ki = 302 nM T32060 CE5QB7 57403569 Ki = 3.8 nM T32060 C68VZL 57403570 Ki = 2.7 nM T32060 CLV07S 57403571 Ki = 1.7 nM T32060 CSWR29 57403903 IC50 = 3180 nM T32060 CWBG94 57403981 Ki > 10000 nM T32060 CQB6F9 57456630 Ki = 22 nM T32060 CQ43XC 57587520 EC50 > 10000 nM T32060 CDG58R 57799306 EC50 = 124 nM T32060 CS6BM2 57799321 Ki = 1796 nM T32060 CUYA69 57799324 Ki = 13 nM T32060 CYPG17 57799326 EC50 > 3000 nM T32060 C0M5PN 57873490 Ki > 1000 nM T32060 CH1BN8 57873491 Ki = 5.1 nM T32060 CI5UO1 57873492 Ki = 164 nM T32060 C2D9HA 57873499 Ki > 1000 nM T32060 C81MLX 57873504 Ki = 69 nM T32060 C7L9IE 57873508 Ki = 28 nM T32060 CZRL39 57873513 Ki = 1000 nM T32060 C98WTS 57873515 Ki = 27 nM T32060 C6BHT3 57873518 Ki = 98 nM T32060 CPX17D 57873520 Ki = 3 nM T32060 C54ROE 57873522 Ki = 40 nM T32060 CM7PI1 57873525 Ki = 50 nM T32060 CMUR21 57873527 Ki = 77 nM T32060 CO5Y9Q 57873531 Ki = 3.6 nM T32060 CHB3D6 58405078 Ki = 225 nM T32060 CX2HU7 58405183 Ki = 5 nM T32060 C3TGM7 58911532 Ki = 275 nM T32060 CFC79Z 58911534 EC50 = 206 nM T32060 CD8JI3 58911579 Ki = 73 nM T32060 CR19FG 58911582 EC50 = 193 nM T32060 C4Z5UB 58911604 Ki = 396 nM T32060 C49INW 58911644 Ki = 2710 nM T32060 CPC3Z0 58911653 Ki = 456 nM T32060 CNEQ36 58911666 Ki = 1081 nM T32060 CJTR58 58911668 Ki = 1424 nM T32060 CG52WR 58911681 EC50 > 2500 nM T32060 C2KP7G 59012632 Ki = 1280 nM T32060 CDX98T 59691557 IC50 = 138 nM T32060 CUAY97 59691584 IC50 = 362 nM T32060 CDB34N 59691661 IC50 = 29 nM T32060 CV8U3A 59691704 IC50 = 91 nM T32060 C1MVB2 59835725 IC50 > 10000 nM T32060 CZ6EF7 59835728 IC50 = 1354 nM T32060 CMG1L8 59835758 IC50 = 1640 nM T32060 CG7JS4 59835780 IC50 = 3290 nM T32060 C42PAO 59835879 IC50 > 10000 nM T32060 C8HYR7 60130337 IC50 = 2330 nM T32060 CYSV60 60165411 Ki = 6982 nM T32060 CB9GC6 60165412 Ki = 204 nM T32060 CI5PM3 60165413 Ki = 3.4 nM T32060 C2Q5VD 60165416 Ki = 132 nM T32060 C9JL3F 60165418 Ki = 224 nM T32060 C31PEN 60165535 Ki = 3812 nM T32060 CP60YF 60165537 Ki > 10000 nM T32060 CP1DR8 60165539 Ki = 1996 nM T32060 C85OTH 60165541 Ki = 287 nM T32060 CJO91V 60165543 Ki = 2206 nM T32060 CJDC53 60165545 Ki > 10000 nM T32060 C3K5JN 60165681 Ki = 523 nM T32060 C5RUP6 60167166 Ki = 36 nM T32060 CRH49P 60167309 Ki = 4255 nM T32060 CX0NY3 60167310 Ki > 10000 nM T32060 COHK72 60167451 Ki = 1548.82 nM T32060 C30SVG 60167452 Ki = 3715.35 nM T32060 CI30FT 60204111 Ki = 311 nM T32060 CWSA08 60204112 Ki = 238 nM T32060 C6AUO2 66800823 Ki = 14 nM T32060 C34ACQ 66800909 Ki = 8.4 nM T32060 CGT9E6 66800910 Ki = 9.5 nM T32060 C0QY7D 66800916 Ki = 6.5 nM T32060 CM58FG 66800926 Ki = 1200 nM T32060 CQ43WD 66800934 Ki = 2.2 nM T32060 CK0I5J 66800939 Ki = 10 nM T32060 C0X2SF 66800942 Ki = 8.8 nM T32060 CFPK92 66800991 Ki = 12 nM T32060 C13GMO 66801000 Ki = 11 nM T32060 CZ1TF9 66801018 Ki = 7.4 nM T32060 CBO9U3 66801028 Ki = 3.8 nM T32060 CA4DM3 66801062 Ki = 0.9 nM T32060 C2OUX9 66801107 Ki = 1.3 nM T32060 C4J5RZ 66801115 Ki = 9.5 nM T32060 C1H8BS 66801116 Ki = 3300 nM T32060 C4JGC6 66801120 Ki = 3.1 nM T32060 CX2GN1 66801139 Ki = 1.6 nM T32060 C1NG8S 66801140 Ki = 15 nM T32060 CR7OW6 66801158 Ki = 0.7 nM T32060 CJU53X 66801160 Ki = 14 nM T32060 CH3BJ8 66801167 Ki = 1.7 nM T32060 C0AV5M 66801173 Ki = 6 nM T32060 C0V9EF 66801186 Ki = 6.5 nM T32060 CTHY41 66801210 Ki = 1 nM T32060 CSD67P 66801225 Ki = 5.7 nM T32060 C8J3YU 66801226 Ki = 98 nM T32060 CX45OZ 66801229 Ki = 0.9 nM T32060 C1S0EV 66801230 Ki = 5.5 nM T32060 C7S1KY 66801234 Ki = 1.5 nM T32060 CB53AV 66801246 Ki = 9.5 nM T32060 C3F1TZ 66801251 Ki = 2.6 nM T32060 CF8O9U 66801259 Ki = 6100 nM T32060 C2Q9FS 66801263 Ki = 10 nM T32060 C7Y9VP 66801267 Ki > 10000 nM T32060 CED17M 66801271 Ki = 5.1 nM T32060 C2FYL1 66801333 Ki = 190 nM T32060 CS75LK 66801335 Ki = 9.5 nM T32060 CDH7S9 66801346 Ki = 2.2 nM T32060 CGC4U6 66801354 Ki = 110 nM T32060 CY4FM5 66801379 Ki = 7.5 nM T32060 C93EGP 66801455 Ki = 8.1 nM T32060 CIRW86 66801551 Ki = 0.7 nM T32060 C8H5PD 66801565 Ki = 9.1 nM T32060 CT5SP8 66801605 Ki = 6.5 nM T32060 C8MH0I 66801613 Ki = 25 nM T32060 C49XBJ 66801673 Ki = 290 nM T32060 C7V8QD 67251061 Ki = 199.53 nM T32060 C1LEH8 67268994 Ki = 187 nM T32060 CI8SB4 67320583 IC50 = 4559 nM T32060 CLA7F3 68281136 Ki = 9.1 nM T32060 C84MZH 68281137 Ki = 210 nM T32060 CWE97U 68490431 Ki > 10000 nM T32060 C6V0RG 68690817 EC50 > 2500 nM T32060 C1R7EY 68691189 EC50 > 2500 nM T32060 C5FAB3 69314950 Ki = 74.1 nM T32060 CKM14W 69432471 Ki = 1 nM T32060 CHKP64 69433076 Ki = 7.7 nM T32060 C5P0ME 69471377 Ki = 4.6 nM T32060 C4FZ6G 69514548 Ki = 1.3 nM T32060 CFND58 69588506 Ki = 2.9 nM T32060 C34GMW 69599704 Ki = 7100 nM T32060 CI16QU 69616387 Ki = 16 nM T32060 CB62XQ 70683433 EC50 = 3020 nM T32060 C6FY2A 70687202 Ki = 55 nM T32060 C9P7YD 70695555 Ki = 430 nM T32060 CVU08A 70695812 Ki > 10000 nM T32060 CYAS63 70697549 EC50 = 9.772 nM T32060 CGXQ60 71041800 IC50 = 1780 nM T32060 CBF6Z8 71109804 Ki = 480 nM T32060 C68NPQ 71109805 Ki = 363 nM T32060 CC43QK 71151588 Ki = 29 nM T32060 C3XNC2 71450247 Ki = 1780 nM T32060 C9VZ8J 71450550 Ki = 1166 nM T32060 C4TWS5 71452172 Ki = 4406 nM T32060 CE0R9D 71454275 Ki = 21570 nM T32060 C8YH0J 71455083 Ki = 54 nM T32060 CAQF34 71455625 Ki > 10000 nM T32060 C6G2HC 71455894 Ki = 4162 nM T32060 C7MNB5 71457264 Ki = 536 nM T32060 CMJ1O9 71457409 Ki = 1825 nM T32060 CP7JI0 71457691 Ki = 3187 nM T32060 C1EA6Q 71458069 Ki = 1.2 nM T32060 CRP65E 71459131 Ki > 1000 nM T32060 CS83IF 71459269 Ki = 810 nM T32060 C5DLQ2 71459553 Ki = 2766 nM T32060 CK5T4P 71459604 Ki = 2259 nM T32060 C63YLA 71461049 Ki = 5962 nM T32060 CJD96I 71461050 Ki > 10000 nM T32060 C5B2WL 71461603 Ki = 1.9 nM T32060 C4P3JU 71462776 Ki = 1019 nM T32060 C3GUQ2 71462777 Ki > 10000 nM T32060 CL91AC 71463022 Ki = 2564 nM T32060 CKX5O8 71463061 Ki = 950 nM T32060 C1DGF4 71499384 IC50 = 75000 nM T32060 CN43VA 71508712 Ki = 89 nM T32060 C2VP0I 71528204 IC50 = 11500 nM T32060 CHY78V 71562549 EC50 > 1000000 nM T32060 CR8Q1X 71562552 EC50 > 1000000 nM T32060 CF4XJ2 71562661 EC50 = 240 nM T32060 C29VZI 71562662 Ki > 300000 nM T32060 CF4BQ7 71562663 Ki > 300000 nM T32060 CRYO82 71562664 EC50 > 1000000 nM T32060 CQ0XA2 71562665 EC50 > 1000000 nM T32060 C5JX3D 71562666 EC50 > 1000000 nM T32060 CR9UC8 71562667 EC50 > 1000000 nM T32060 C9EIY7 71566778 IC50 = 1300 nM T32060 CT2ME3 71574204 Ki = 90 nM T32060 C3SXR5 71574206 Ki = 115 nM T32060 C2YRI9 71574208 Ki = 65 nM T32060 C62RWV 71574210 Ki = 47 nM T32060 CKC53S 71574212 Ki = 34 nM T32060 CNV42M 71574298 Ki = 42 nM T32060 C9PGQ1 71574300 Ki = 23 nM T32060 C2LXH5 71574302 Ki = 22 nM T32060 C2YPB8 71574304 Ki = 29 nM T32060 CK7GM0 71574306 Ki = 35 nM T32060 C5LY9W 71681897 Ki = 337 nM T32060 CG34PR 71681898 Ki = 1460 nM T32060 CG4V0A 71682216 Ki = 1448 nM T32060 CI46CW 71682217 Ki = 231 nM T32060 C61JZW 71691223 Ki = 1359.45 nM T32060 C0W2YA 71727193 Ki = 2182 nM T32060 C6CIB5 71727196 Ki = 561 nM T32060 CQO30I 71733932 Ki = 28000 nM T32060 C93QMB 71733935 Ki = 9000 nM T32060 C53MXL 71815503 IC50 = 205 nM T32060 CF01OQ 71937057 Ki = 33 nM T32060 C0PSF9 72138721 Ki = 99 nM T32060 CR3Z1P 72152555 Ki = 136 nM T32060 C24ZSV 72152556 Ki = 102 nM T32060 CWT8O4 72152557 Ki = 29 nM T32060 CZ49CG 72152558 Ki > 10000 nM T32060 C3ATN5 72197484 EC50 = 6.1 nM T32060 C20HSN 72197485 EC50 = 27.9 nM T32060 CN8A5R 72197486 IC50 = 3 nM T32060 CL3BF7 72197668 EC50 = 77.6 nM T32060 CUVJ59 72197845 Ki = 71 nM T32060 CIKU20 72198011 Ki = 498 nM T32060 CWH6T3 72548703 IC50 = 0.64 nM T32060 C80VRM 72549033 Ki = 123 nM T32060 C8Z0NM 72550642 Ki = 478 nM T32060 CL6W2Q 72550645 Ki = 77 nM T32060 C78LYM 72698087 Ki > 10000 nM T32060 C63HPK 72698088 Ki = 8700 nM T32060 C4AS0E 72699528 Ki = 0.28 nM T32060 CO20CN 72699532 Ki = 8.1 nM T32060 C8EVJ6 72699690 Ki = 0.26 nM T32060 CEAK86 72699692 Ki = 0.6 nM T32060 COH4F8 72699779 Ki = 3.2 nM T32060 C26STM 72700473 Ki = 5.8 nM T32060 CL96GC 72700475 Ki = 0.63 nM T32060 C45JKS 72700476 Ki = 0.36 nM T32060 C3TO8B 72700557 Ki = 0.24 nM T32060 CVA2X7 72700634 Ki = 0.29 nM T32060 C7W4RH 72734860 Ki = 1000 nM T32060 CC6Q5R 72771081 Ki < 100 nM T32060 CC65OA 73213195 Ki = 736 nM T32060 CW83DK 73213196 Ki = 257 nM T32060 C0QCH3 73345916 IC50 = 2753 nM T32060 C2N9RL 73345917 IC50 = 4578 nM T32060 CCNF45 73345918 IC50 > 10000 nM T32060 C6K8QF 73345919 IC50 = 947 nM T32060 C9SN7B 73345920 IC50 = 2084 nM T32060 CCV91B 73346042 Ki > 10000 nM T32060 CK0HR9 73346334 Ki > 10000 nM T32060 CXM8O2 73347306 IC50 = 950 nM T32060 C9X8GY 73347307 IC50 = 1000 nM T32060 C8LUG4 73347433 IC50 > 10000 nM T32060 C9GWD1 73347434 IC50 > 10000 nM T32060 CJ93GA 73347436 IC50 = 25.1 nM T32060 C3LO5H 73347437 IC50 = 28.8 nM T32060 C1FE6O 73347438 IC50 > 10000 nM T32060 CTG14R 73347439 IC50 = 6577 nM T32060 C8TCG6 73347440 IC50 = 17.9 nM T32060 CJP8E5 73347441 IC50 = 696 nM T32060 CFW96K 73347828 Ki > 10000 nM T32060 CAZ9C2 73348087 IC50 = 175 nM T32060 C9RQM2 73348967 IC50 = 57.4 nM T32060 C5QDC1 73348968 IC50 = 3666 nM T32060 C4XAH0 73348969 IC50 = 4535 nM T32060 CJGF08 73348970 IC50 = 2198 nM T32060 CV31UL 73348972 IC50 = 9.1 nM T32060 CW8A0Y 73349359 Ki = 3060 nM T32060 C6BS5L 73349361 Ki = 1732 nM T32060 CY2IB5 73349362 Ki > 10000 nM T32060 C2CO5J 73350529 EC50 = 2900 nM T32060 C3B9NI 73350530 IC50 > 10000 nM T32060 C96DHM 73350531 IC50 > 10000 nM T32060 CZ7A4S 73350532 IC50 = 4499 nM T32060 C6LTU4 73350533 IC50 = 1268 nM T32060 CA20WC 73350534 IC50 = 5866 nM T32060 CKLH28 73350535 IC50 = 3673 nM T32060 CC8I7X 73351903 IC50 > 1000 nM T32060 CG4M8P 73351905 IC50 > 1000 nM T32060 CZTE85 73352046 EC50 = 687 nM T32060 CXZY13 73352047 IC50 = 2625 nM T32060 C6ZGY5 73352048 EC50 = 153 nM T32060 C0FWE9 73352049 IC50 = 27.2 nM T32060 CE09NW 73353508 IC50 > 10000 nM T32060 CRZ64E 73353509 IC50 = 684 nM T32060 CQOZ67 73353510 IC50 = 1894 nM T32060 CZ5C3G 73353511 IC50 > 10000 nM T32060 CX4Q8N 73353512 IC50 = 4880 nM T32060 CBN58Q 73353513 IC50 = 350 nM T32060 CAR7Z5 73354882 IC50 = 400 nM T32060 CY8S2M 73354999 IC50 > 10000 nM T32060 CN0P6A 73355000 EC50 = 1200 nM T32060 C23EYP 73355001 IC50 > 10000 nM T32060 CXM09L 73355002 IC50 > 10000 nM T32060 C61AQJ 73355003 EC50 = 96.3 nM T32060 CVFM82 73355005 IC50 > 10000 nM T32060 CNQ69I 73355006 IC50 = 5283 nM T32060 CQSJ15 73355007 IC50 = 163 nM T32060 CQZW41 73355008 IC50 = 52.2 nM T32060 CET52A 73356443 IC50 > 1000 nM T32060 CQAO31 73356563 IC50 = 1.95 nM T32060 CA6L7B 73356564 IC50 = 9741 nM T32060 C2E7QW 75201901 Ki = 4900 nM T32060 C8IDL3 75306277 Ki = 1.995 nM T32060 CS3HT5 76309671 Ki = 1548.82 nM T32060 C69BJY 76310154 Ki = 19.05 nM T32060 CN52QU 76310158 Ki = 42.66 nM T32060 CTV52G 76313854 Ki = 31.62 nM T32060 CP40AM 76313855 Ki = 63.1 nM T32060 C3B8FS 76313862 Ki = 794.33 nM T32060 CQP0O8 76317383 Ki = 4.467 nM T32060 C6WXK7 76319003 Ki = 22540 nM T32060 CE5C2B 76319004 Ki = 125.89 nM T32060 C2NXG0 76321107 Ki = 5.012 nM T32060 C5TQ0X 76322648 Ki = 330.37 nM T32060 CNZQ23 76324322 Ki = 1.1 nM T32060 CW7RV4 76324757 Ki = 630.96 nM T32060 CQ8D4Y 76324758 Ki = 512.86 nM T32060 C8SOZ7 76328295 Ki = 10.96 nM T32060 C5M8OD 76328296 Ki = 6.607 nM T32060 CTL3I7 76331989 Ki = 15.85 nM T32060 C9KVC1 76333484 Ki = 307.5 nM T32060 CGBE87 76335066 Ki = 5.1 nM T32060 CUO0S5 76335562 Ki = 23.44 nM T32060 CL41EG 76335563 Ki = 158.49 nM T32060 C28RIZ 76518514 Ki = 317 nM T32060 C70ZVB 86221574 Ki = 5693 nM T32060 CJ9N5Q 86280005 Ki = 0.33 nM T32060 CCY5N2 86302554 Ki = 3100 nM T32060 CUA89I 86341962 Ki = 0.18 nM T32060 CWPH45 86341996 Ki = 0.21 nM T32060 CCR8X7 86342061 Ki = 0.14 nM T32060 CY2I8J 86342094 Ki = 0.35 nM T32060 CC47HJ 86342098 Ki = 0.91 nM T32060 CK03YC 86342156 Ki = 0.19 nM T32060 C5AQK2 86342192 Ki = 0.15 nM T32060 C9DZ2I 86342193 Ki = 0.29 nM T32060 CQP38R 86342194 Ki = 0.64 nM T32060 CE39OD 86342294 Ki = 0.3 nM T32060 CP76JG 88912137 Ki = 605 nM T32060 CG9CM0 89750383 IC50 = 356 nM T32060 CD7R6P 90213677 Ki = 0.21 nM T32060 CFDW68 90644074 Ki = 4200 nM T32060 C0T8RE 90644075 Ki = 950 nM T32060 C2KE9G 90644076 Ki = 970 nM T32060 C1SOF5 90644077 Ki = 410 nM T32060 CIE9Z2 90644078 Ki = 63 nM T32060 CLFV10 90644226 Ki = 22 nM T32060 CZ7LD8 90644227 Ki = 16 nM T32060 C35GPQ 90644228 Ki = 56 nM T32060 CZI30L 90644230 Ki = 81 nM T32060 CWMU25 90644511 IC50 = 360 nM T32060 CVG2C1 90654672 Ki = 2010 nM T32060 C2EZX4 90655112 Ki = 14 nM T32060 C6EZ3G 90655113 Ki = 1.7 nM T32060 CA08SW 90655114 Ki = 14 nM T32060 C42ELK 90655115 Ki = 5.8 nM T32060 C51ZIC 90655116 Ki > 1000 nM T32060 C4JOT3 90655117 Ki = 671 nM T32060 CK3D1X 90655118 Ki = 18 nM T32060 CG2VY6 90655119 Ki = 50 nM T32060 CV4H2G 90655120 Ki > 1000 nM T32060 CUJQ70 90655121 Ki = 702 nM T32060 CL3RP6 90655122 Ki > 1000 nM T32060 C2P0LK 90655123 Ki > 1000 nM T32060 CVQC46 90655124 Ki > 1000 nM T32060 CB4Y0S 90655125 Ki = 324 nM T32060 CH8YX5 90655126 Ki = 5.5 nM T32060 C8XT6K 90655127 Ki = 17 nM T32060 C98YWT 90655128 Ki = 5.2 nM T32060 CBI6Y5 90664323 IC50 = 95 nM T32060 C2PV7O 90664324 IC50 = 20 nM T32060 CO4V5L 90664325 IC50 = 5.17 nM T32060 C2RW9Y 90664326 IC50 = 13 nM T32060 C6T1KX 90664327 IC50 = 16.8 nM T32060 C81IBN 90664328 IC50 = 21 nM T32060 C75ZUE 90664329 IC50 = 318 nM T32060 CM7HQ9 90664330 IC50 = 8.63 nM T32060 CA2BO3 90664449 IC50 = 94 nM T32060 C9ULV4 90664450 IC50 = 19.5 nM T32060 CH02GV 90664451 IC50 = 70.9 nM T32060 CIL2W9 90664452 IC50 = 12.3 nM T32060 C7RT9G 90664453 IC50 = 52.1 nM T32060 C3AX1O 90664454 IC50 = 45.5 nM T32060 CPGI68 90664459 IC50 = 67 nM T32060 CICD63 90664460 IC50 = 20 nM T32060 CBZT19 90664586 IC50 = 196 nM T32060 C5HRY0 90664587 IC50 = 107 nM T32060 CG6V1D 90664589 IC50 = 104 nM T32060 C7W5SH 90664590 IC50 = 106 nM T32060 CNU6J8 90664598 IC50 = 29 nM T32060 CB95PE 90664599 IC50 = 24 nM T32060 CA68PB 90664600 IC50 = 27 nM T32060 C4MUI2 90664601 IC50 = 18.6 nM T32060 CA79EY 90664683 IC50 = 43 nM T32060 CHY82Q 90664697 IC50 = 275.1 nM T32060 CM0Y7P 90664699 IC50 = 139 nM T32060 CEF0R5 90664700 IC50 = 171 nM T32060 CR07QH 90664701 IC50 = 23.1 nM T32060 CZ69VH 90664702 IC50 = 197 nM T32060 CF4P3I 90664703 IC50 = 254 nM T32060 CR7LX6 90664705 IC50 = 63.1 nM T32060 CNT10P 90664709 IC50 = 80 nM T32060 C35BTL 90664710 IC50 = 39 nM T32060 CDPV60 90664712 IC50 = 21 nM T32060 CG7D2H 90664713 IC50 = 55 nM T32060 CZJN57 90664814 IC50 = 176.6 nM T32060 CR87PO 90664815 IC50 = 54 nM T32060 CN7W8A 90664816 IC50 = 30 nM T32060 CI8B6Q 90664817 IC50 = 26.7 nM T32060 CEN36Q 90664818 IC50 = 40 nM T32060 CJ73WT 90664819 IC50 = 237 nM T32060 C5AWS4 90664820 IC50 = 97.6 nM T32060 CL3AW1 90664821 IC50 = 170 nM T32060 C1C2HB 90664822 IC50 = 154 nM T32060 CQ4T3E 90664830 IC50 = 32.4 nM T32060 CKM05S 90664904 IC50 > 10000 nM T32060 CTR58M 90664931 IC50 = 58 nM T32060 CP9SI1 90664949 IC50 = 58 nM T32060 CZ19LO 90664951 IC50 = 15.2 nM T32060 CLN9K2 90664952 IC50 = 38 nM T32060 CO5Y3C 90664958 IC50 = 90 nM T32060 C74XDT 90664959 IC50 = 28 nM T32060 CWQ18M 90664960 IC50 = 201 nM T32060 C07WIP 90664961 IC50 = 57 nM T32060 CHT7D5 90664962 IC50 = 31 nM T32060 C04UEP 90665072 IC50 = 147 nM T32060 CF90MU 90665073 IC50 = 127 nM T32060 C8YX4R 90665074 IC50 = 12.2 nM T32060 CP5QO8 90665075 IC50 = 20.1 nM T32060 C3XIQ2 90665076 IC50 = 80.6 nM T32060 CI8JU1 90665077 IC50 = 12.8 nM T32060 C67AXN 90665078 IC50 = 21 nM T32060 CQ95OT 90665079 IC50 = 56 nM T32060 C7JLM9 90665080 IC50 = 582 nM T32060 CZHA09 90665086 IC50 = 96.8 nM T32060 C17EWV 90665087 IC50 = 47 nM T32060 CO46PW 90665091 IC50 = 26 nM T32060 CXJ62T 90665173 IC50 = 21 nM T32060 CYD25E 90665193 IC50 = 9.86 nM T32060 CG98QO 90665194 IC50 = 13.9 nM T32060 C5PN4D 90665195 IC50 = 182.1 nM T32060 C7XIS2 90665197 IC50 = 370 nM T32060 CIJ5M0 90665200 IC50 = 48 nM T32060 C09JPN 90665201 IC50 = 14.2 nM T32060 C8BV5P 90665202 IC50 = 10.3 nM T32060 C9JQ8U 90666896 Ki = 10 nM T32060 CKY24S 90666897 Ki = 125.89 nM T32060 CVI58C 90666898 Ki = 19.95 nM T32060 CACG19 90666899 Ki = 5.012 nM T32060 C4HPT5 90666900 Ki = 79.43 nM T32060 C8DM7O 90666901 Ki = 281.84 nM T32060 C86HDZ 90666902 Ki = 19.95 nM T32060 CODM50 90666903 Ki = 7.943 nM T32060 CSN13Z 90666904 Ki = 39.81 nM T32060 CSRU41 91242334 IC50 = 683 nM T32060 CRX16J 91884611 IC50 = 2.9 nM T32060 CDWS84 91937906 Ki = 2831 nM T32060 C3K4LU 91937908 Ki = 264 nM T32060 CUQ6V0 92042918 EC50 = 374 nM T32060 CGC29J 92042920 EC50 = 359 nM T32060 CLR87F 94496003 Ki = 55 nM T32060 CNUM64 95104704 Ki = 2268 nM T32060 CK83CL 95198280 Ki = 934 nM T32060 CMG1N3 95214051 Ki = 4049 nM T32060 C5GJA7 95232163 Ki = 1443 nM T32060 C8QJW7 95338888 Ki = 423 nM T32060 C0BAG2 95339350 Ki = 3474 nM T32060 C4BRK3 95339542 Ki = 282 nM T32060 C8XFV3 101007561 Ki = 275 nM T32060 C02GRK 104697662 Ki > 10000 nM T32060 CG6W0P 112485369 EC50 = 249 nM T32060 CP6F4D 112815120 Ki = 171 nM T32060 C8V2SN 116887744 EC50 > 10000 nM T32060 CP0I7M 117887098 IC50 = 6200 nM T32060 CM78SL 118335021 IC50 = 650 nM T32060 CK83OB 118335025 IC50 = 2300 nM T32060 CEMZ15 118464420 Ki = 211 nM T32060 CV2L6O 118464425 Ki = 1541 nM T32060 CFNG86 118464427 Ki = 1313 nM T32060 CMSN80 118626035 Ki = 36 nM T32060 CT3AI0 118626042 Ki = 82 nM T32060 CKNJ72 118626045 Ki = 9 nM T32060 CGB42Y 118626088 Ki = 296 nM T32060 C0XJT5 118626089 Ki = 9 nM T32060 CIE4C7 118626101 Ki = 76 nM T32060 C1NYS5 118626120 Ki = 91 nM T32060 CPG04R 118626121 Ki = 19 nM T32060 C3S5LJ 118626129 Ki = 56 nM T32060 CY3F0N 118626140 Ki = 238 nM T32060 CE07IQ 118626142 Ki = 26 nM T32060 C72OZY 118626161 Ki = 21 nM T32060 CY3E7S 118626169 Ki = 390 nM T32060 CHRB75 118626208 Ki = 110 nM T32060 CF5K0V 118691439 Ki = 37.3 nM T32060 CW15HU 118700678 Ki > 9300 nM T32060 CSB25E 118709750 Ki = 509 nM T32060 CD4S9R 118709751 Ki = 115 nM T32060 CO8E9F 118711252 Ki > 1000 nM T32060 CJY9D7 118711253 Ki > 1000 nM T32060 CFJE45 118711254 Ki = 4.52 nM T32060 CK1A2W 118711255 Ki = 10.3 nM T32060 CNQJ96 118711256 Ki = 9.95 nM T32060 CJ91QY 118711257 Ki = 192 nM T32060 C42YEC 118711258 Ki = 862 nM T32060 CX3M2Z 118711262 Ki = 163 nM T32060 CW3F4T 118711265 Ki = 826 nM T32060 C9Z3PH 118713118 EC50 = 246 nM T32060 CUV5Y0 118715454 EC50 > 30000 nM T32060 C5LFW4 118717221 Ki > 1000 nM T32060 CES97Y 118722639 Ki = 18 nM T32060 CM3P7R 118722912 Ki = 1228 nM T32060 CP3QC2 118722913 Ki = 11 nM T32060 C1PG3C 118722914 Ki = 8 nM T32060 CR6E5D 118722915 Ki = 17 nM T32060 CE05XG 118727442 IC50 = 329 nM T32060 C1ZH2I 118727443 IC50 = 702 nM T32060 C0M5AR 118727444 IC50 = 247 nM T32060 CDHS51 118727445 IC50 = 253 nM T32060 CWZ7P0 118727447 IC50 = 479 nM T32060 CH9V1A 118727448 IC50 = 1593 nM T32060 C6AZG2 118727449 IC50 = 555 nM T32060 CZ1LD0 118727450 IC50 = 433 nM T32060 CU3X0M 118729231 Ki = 370 nM T32060 CNE49D 118729233 Ki = 20 nM T32060 CLD1Z7 118729234 Ki = 80 nM T32060 C4RDW3 118729235 Ki = 1100 nM T32060 C47XHR 118729237 Ki = 760 nM T32060 C08FQG 118729239 Ki = 8100 nM T32060 CR0HA4 118729241 Ki = 2000 nM T32060 CY36XK 118729243 Ki = 210 nM T32060 C1VK9B 118729245 Ki = 220 nM T32060 CVR67P 118729247 Ki = 60 nM T32060 CA2Y1F 118729249 Ki = 250 nM T32060 CE1IB3 118729250 Ki = 50 nM T32060 CI8WR2 118729251 Ki = 140 nM T32060 C4ML5K 118729252 Ki = 71 nM T32060 COCH98 118729253 Ki = 74 nM T32060 CQ7K5G 118729255 Ki = 500 nM T32060 C2LDI1 118729257 Ki = 80 nM T32060 COQ04B 118729259 Ki = 1300 nM T32060 C9BG0R 118729261 Ki = 20 nM T32060 C63GWU 118729262 Ki = 260 nM T32060 CN24KA 118729263 Ki = 40 nM T32060 C7ZJ2F 118729265 Ki = 130 nM T32060 CL5W0J 118729267 Ki = 110 nM T32060 CN65HD 118729269 Ki = 320 nM T32060 C2B6YA 118729271 Ki = 30 nM T32060 CZ40RY 118729273 Ki = 650 nM T32060 CE38GM 118729275 Ki = 44 nM T32060 CS9W7L 118729277 Ki = 2800 nM T32060 C9LI7N 118729278 Ki = 2400 nM T32060 C8TEX7 118729279 Ki = 700 nM T32060 CW3R9X 118729280 Ki = 1000 nM T32060 C5O2NU 118729733 Ki = 18130 nM T32060 CTE58Z 118730369 Ki = 500 nM T32060 CD21PC 118731187 IC50 = 6000 nM T32060 CSW75A 118731193 IC50 = 5200 nM T32060 C8GKX6 118731351 Ki = 166 nM T32060 CQ8F6C 118731354 Ki = 2148 nM T32060 CU12XM 118731356 Ki = 1684 nM T32060 CJ1VX4 118733762 EC50 = 1215 nM T32060 CQZ71R 118733794 EC50 = 1005 nM T32060 C7ZS0V 118733802 EC50 = 903 nM T32060 C6VO5G 118733806 EC50 = 1476 nM T32060 C7RUF2 118733808 EC50 = 1305 nM T32060 CNH6K2 118733810 EC50 = 1811 nM T32060 CSN70M 118733818 EC50 = 1025 nM T32060 CD3E4N 118733819 EC50 = 697 nM T32060 CC4G2U 118733823 EC50 = 1666 nM T32060 C98ZTE 118733825 EC50 = 2994 nM T32060 C5RNW2 118857804 Ki = 2380 nM T32060 C0GQF1 118857828 Ki > 10000 nM T32060 C6UHM8 118857829 Ki > 10000 nM T32060 CA03SM 118857831 Ki > 10000 nM T32060 C0FCX2 118857833 Ki > 10000 nM T32060 CU1Z8O 118857834 Ki > 10000 nM T32060 CX2RY8 118857835 Ki > 10000 nM T32060 C2ZD0T 118857837 Ki > 10000 nM T32060 CB54AQ 118857838 Ki > 10000 nM T32060 CHJ70O 118960212 IC50 = 240 nM T32060 C35WTP 122177641 Ki = 8000 nM T32060 C8OS7B 122177642 Ki = 14000 nM T32060 CV2AT4 122177644 Ki = 1000 nM T32060 CB16GY 122177645 Ki = 710 nM T32060 C7W3EY 122178698 Ki = 818 nM T32060 CF8P1H 122178699 Ki = 268 nM T32060 C48MFR 122178700 Ki = 239 nM T32060 CZ72QS 122178701 Ki = 570 nM T32060 C4VY8A 122178702 Ki = 1156 nM T32060 C2KF4Z 122178703 Ki = 750 nM T32060 CX6MJ2 122178704 Ki = 377 nM T32060 CA53KF 122178705 Ki = 244 nM T32060 C8XD3F 122178706 Ki = 446 nM T32060 CTRC59 122178707 Ki = 582 nM T32060 C5QV8D 122178708 Ki = 570 nM T32060 C84UED 122178709 Ki = 383 nM T32060 CV96JK 122178710 Ki = 216 nM T32060 CM89KS 122178711 Ki = 418 nM T32060 CH9SX5 122180956 Ki = 510 nM T32060 C2LW4N 122180957 Ki = 0.6026 nM T32060 CM1EW3 122180958 Ki = 0.6026 nM T32060 C3LJ8I 122180959 Ki = 1.698 nM T32060 C4NA2C 122180960 Ki = 10.96 nM T32060 CP7DG4 122180961 Ki = 0.1995 nM T32060 C6P9QO 122180962 Ki = 7.762 nM T32060 C8DSW3 122180963 Ki = 12.02 nM T32060 CS63HY 122180964 Ki = 12.88 nM T32060 CU4X9I 122180966 Ki = 79.43 nM T32060 CXQ4C1 122180967 Ki = 38.9 nM T32060 CX1N4V 122180968 Ki = 83.18 nM T32060 C90BHR 122180969 Ki = 141.25 nM T32060 CIL05K 122180970 Ki = 3.09 nM T32060 C0F9UN 122180971 Ki = 19.95 nM T32060 C2H8CK 122180972 Ki = 30.9 nM T32060 CKJ21N 122180973 Ki = 316.23 nM T32060 C6GI9R 122180974 Ki = 3.311 nM T32060 CBS6G1 122180975 Ki = 0.1995 nM T32060 CDT10B 122180976 Ki = 0.4365 nM T32060 C6A4CD 122180977 Ki = 1.349 nM T32060 CCV9D5 122181326 Ki = 540 nM T32060 C5D1NC 122181329 Ki = 89 nM T32060 C05RGV 122181330 Ki = 550 nM T32060 C3XGN0 122181333 Ki = 210 nM T32060 CXL5V3 122183764 Ki = 2.4 nM T32060 CK3VT8 122183765 Ki = 1.7 nM T32060 C12TRH 122183771 Ki = 55 nM T32060 C06GQO 122183778 Ki = 350 nM T32060 CTJO50 122184561 IC50 = 360 nM T32060 CZ1MA3 122184562 IC50 > 10000 nM T32060 CH37IW 122184563 IC50 = 528 nM T32060 C5JTD9 122184564 IC50 = 8150 nM T32060 CJR48E 122184670 IC50 = 646 nM T32060 C7YA0Q 122184671 IC50 = 138 nM T32060 C6RP0N 122184672 IC50 = 34 nM T32060 CLP36J 122184673 IC50 = 1460 nM T32060 C5Y0KX 122184691 IC50 = 4540 nM T32060 C18ZKO 122184692 IC50 > 10000 nM T32060 C0XJK1 122184693 IC50 > 10000 nM T32060 C97APV 122184694 IC50 > 10000 nM T32060 CLK94O 122184695 IC50 > 10000 nM T32060 CWSF63 122184696 IC50 > 10000 nM T32060 CW8L5K 122184697 IC50 > 10000 nM T32060 CI4SF6 122184698 IC50 = 595 nM T32060 CDHE98 122184699 IC50 = 790 nM T32060 CIU9W5 122184700 IC50 > 10000 nM T32060 CU2PG6 122184701 IC50 = 1410 nM T32060 CKG74I 122184702 IC50 > 10000 nM T32060 CZ0I1K 122184703 IC50 = 242 nM T32060 C65COE 122184704 IC50 = 713 nM T32060 CHS9N7 122184705 IC50 > 10000 nM T32060 CWM9Q7 122184706 IC50 = 9650 nM T32060 CHV3U1 122187388 Ki = 120.13 nM T32060 CW4H5Y 122187389 Ki = 109.17 nM T32060 C4FUN7 122187390 Ki = 92.05 nM T32060 C98GZL 122187391 Ki = 383.02 nM T32060 CJQT21 122187392 Ki = 145.64 nM T32060 CI7F8R 122187393 Ki = 149.11 nM T32060 C7CW3P 122187394 Ki = 65.78 nM T32060 CR0H6S 122187395 Ki = 267.7 nM T32060 CA25FV 122187396 Ki = 83.38 nM T32060 CI6NK0 122187397 Ki = 45.77 nM T32060 CY2JF0 122187398 Ki = 69.99 nM T32060 C90DZQ 122187399 Ki = 14.04 nM T32060 C94UQF 122187400 Ki = 496.24 nM T32060 C0UDY2 122187401 Ki = 42.14 nM T32060 COFU75 122187402 Ki = 234.77 nM T32060 CU1FI9 122187403 Ki = 184.33 nM T32060 CK5BP3 122189387 Ki = 84 nM T32060 C8JV3W 122189388 Ki = 6.9 nM T32060 CV1U4Q 122189389 Ki = 15 nM T32060 C4PBA3 122189390 Ki = 50 nM T32060 CD7UN3 122189391 Ki = 89 nM T32060 C14FCX 122189392 Ki = 7.1 nM T32060 C1NIK8 122189393 Ki = 5.3 nM T32060 C9KXH4 122189394 Ki = 0.64 nM T32060 CBHT01 122377930 Ki = 178 nM T32060 CLW53P 122483274 Ki = 257 nM T32060 CO63ET 122483280 Ki = 451 nM T32060 C4QM2E 124247485 Ki = 175 nM T32060 CM57GR 126720252 Ki = 8400 nM T32060 CLWM12 126720394 Ki = 449 nM T32060 C8Q1JB 126720403 Ki = 475 nM T32060 C1U3SZ 126720425 Ki = 694 nM T32060 C5G8FD 126720440 Ki = 441 nM T32060 CCM0S8 126844990 EC50 = 3679 nM T32060 CIHZ54 127025242 Ki = 1297 nM T32060 CCY7P3 127025243 Ki = 1295 nM T32060 CTBN56 127026052 Ki = 245.47 nM T32060 CTYP30 127026133 Ki = 1146 nM T32060 CBE56W 127026514 Ki = 1265 nM T32060 CAX87V 127026556 EC50 = 2332 nM T32060 CX6EI2 127026750 Ki = 303 nM T32060 CH9JB5 127026860 EC50 = 949 nM T32060 CU29SR 127027463 EC50 = 1071.52 nM T32060 CW40RC 127028088 EC50 = 436.52 nM T32060 C7A8OC 127028095 EC50 = 67.61 nM T32060 CI1SF6 127028096 EC50 = 933.25 nM T32060 CGA51D 127028100 EC50 = 20.89 nM T32060 C90QPM 127028101 EC50 = 119 nM T32060 CALC05 127028403 EC50 = 426 nM T32060 C0SGM2 127028405 EC50 = 81 nM T32060 CE0T8G 127028406 EC50 = 81 nM T32060 C3H9NU 127028407 EC50 = 361 nM T32060 C8MC1I 127028408 EC50 = 489.78 nM T32060 CBU65F 127028421 EC50 = 92 nM T32060 C9YU1E 127028422 EC50 = 165.96 nM T32060 CPF1T5 127028423 EC50 = 17.78 nM T32060 CA9IP6 127028732 EC50 = 794.33 nM T32060 CC4U8R 127029581 EC50 = 645.65 nM T32060 C6O2SL 127034715 Ki = 146 nM T32060 CNO80F 127034729 Ki = 1507 nM T32060 CB02LG 127034730 Ki = 2234 nM T32060 CZ61LK 127034966 EC50 > 5011.87 nM T32060 CA0SN5 127034967 EC50 > 5011.87 nM T32060 CQ0ZT9 127035062 Ki = 165 nM T32060 CW1KD7 127035063 Ki = 140 nM T32060 CO3W6A 127035064 Ki = 200 nM T32060 CTY04X 127035065 Ki = 267 nM T32060 CPM2B8 127035066 Ki = 919 nM T32060 CU49VE 127036186 Ki = 724.44 nM T32060 CP04WI 127036910 Ki = 3531 nM T32060 CG06BD 127036932 Ki = 407.38 nM T32060 CVW71O 127036953 Ki = 478.63 nM T32060 C0HLY8 127037059 Ki = 226 nM T32060 CZ6QR4 127037093 Ki = 1472 nM T32060 C2XBE8 127037921 Ki = 1479 nM T32060 CX0CN4 127037922 Ki = 70 nM T32060 C8TC9G 127038281 Ki = 30 nM T32060 CYJ2D5 127039593 Ki = 378 nM T32060 C8D4AV 127040908 Ki = 382 nM T32060 C15BGV 127041244 Ki = 264 nM T32060 CU0J4S 127041258 Ki = 230 nM T32060 C20MZH 127041259 Ki = 121 nM T32060 CP16CZ 127041260 Ki = 1254 nM T32060 CZT53S 127041261 Ki = 1928 nM T32060 C0FJP2 127041563 Ki = 1070 nM T32060 CUC3F9 127041564 Ki = 557 nM T32060 COG9D2 127041874 Ki = 42 nM T32060 CS4WH1 127042184 Ki = 69 nM T32060 C13AIN 127042185 Ki = 58 nM T32060 CR59TP 127042539 Ki = 429 nM T32060 C54IZC 127042540 Ki = 413 nM T32060 C8G1HF 127042841 Ki = 1328 nM T32060 CS9V0E 127048333 Ki = 65 nM T32060 CQM81O 127048334 Ki = 43 nM T32060 CJG5E2 127048335 Ki = 54 nM T32060 CUK40V 127048336 Ki = 75 nM T32060 C0V5YU 127048532 IC50 = 1320 nM T32060 CHW0L2 127048533 IC50 = 720 nM T32060 C9QR6V 127048539 IC50 = 80 nM T32060 CU6K4P 127048540 IC50 = 1900 nM T32060 C42FHY 127049060 Ki = 977.24 nM T32060 CF2QY9 127049061 Ki > 10000 nM T32060 CN2F1W 127049163 IC50 > 10000 nM T32060 C1TI6J 127049515 IC50 = 360 nM T32060 CT16PL 127049516 IC50 = 860 nM T32060 C4QKS3 127049517 IC50 = 840 nM T32060 C03BLH 127049522 IC50 = 2200 nM T32060 C2IX7Q 127049847 IC50 = 340 nM T32060 CRK8W3 127049848 IC50 = 1400 nM T32060 C85PIF 127049849 IC50 = 494 nM T32060 CO2V5Z 127049850 IC50 = 1380 nM T32060 C27MWC 127049861 IC50 = 820 nM T32060 CZS1L6 127049862 IC50 = 46 nM T32060 CZD91J 127049863 IC50 = 15 nM T32060 C1S6EN 127049864 IC50 = 180 nM T32060 C2H0BQ 127049865 IC50 = 35 nM T32060 CUK1S9 127049866 IC50 = 216 nM T32060 C6SP9O 127049979 Ki = 365 nM T32060 C1CB0Z 127049980 Ki = 221 nM T32060 C0JUA9 127049981 Ki = 288 nM T32060 C69RCG 127049982 Ki = 185 nM T32060 C0M9PE 127049983 Ki = 125 nM T32060 CI5XG2 127050282 Ki = 103 nM T32060 CX53AC 127050632 Ki = 1123 nM T32060 CP9UT4 127050764 IC50 = 1050 nM T32060 C9T2VY 127050765 IC50 = 1100 nM T32060 CIOZ65 127051038 IC50 = 1100 nM T32060 C7XK3G 127051039 IC50 = 670 nM T32060 CR4TV6 127051040 IC50 = 1100 nM T32060 CCTO35 127051041 IC50 = 460 nM T32060 CA2SJ6 127051340 IC50 = 30.3 nM T32060 CX5H1W 127051482 Ki = 185 nM T32060 CTL0S1 127051516 Ki > 10000 nM T32060 CTL8J1 127051843 Ki = 22.91 nM T32060 CF6V9Q 127051844 Ki = 404 nM T32060 C8TNB1 127051845 Ki = 2137.96 nM T32060 CT9O7G 127051863 Ki = 5970 nM T32060 C5ONG1 127051864 Ki > 10000 nM T32060 CRF85X 127052458 Ki = 724.44 nM T32060 CCY71I 127052465 Ki > 10000 nM T32060 C2E9VX 127052467 Ki = 926 nM T32060 CPO4C3 127052468 Ki = 522.5 nM T32060 CSQ2N8 127052486 Ki = 3388.44 nM T32060 CT9RS4 127052488 Ki = 519 nM T32060 CLU7C1 127052757 Ki = 726 nM T32060 C95KYT 127052758 Ki = 322 nM T32060 CYNR02 127052759 Ki = 317 nM T32060 C14YJU 127052778 Ki = 1071.52 nM T32060 C1JAS7 127052779 Ki = 165.96 nM T32060 C6XR8U 127053028 Ki = 169 nM T32060 C7MQK8 127053042 Ki = 1778.28 nM T32060 C3WIA6 129103318 IC50 = 257.4 nM T32060 CBX2V6 129186527 IC50 = 9.49 nM T32060 CV2K7I 129186528 IC50 = 12.2 nM T32060 CD9C1F 129186530 IC50 = 1110 nM T32060 C2F5YE 129186531 IC50 = 814 nM T32060 C6GC0F 129186534 IC50 = 10.2 nM T32060 CTP0O3 129186549 IC50 = 7.66 nM T32060 C8KM6N 129186554 IC50 = 1.19 nM T32060 C7FR6U 129186558 IC50 = 65.4 nM T32060 CEZT92 129186564 IC50 = 11.5 nM T32060 CT4P7U 129718902 Ki > 10000 nM T32060 C1CV2Y 129840786 Ki = 112 nM T32060 CJ5S2O 129840806 Ki > 10000 nM T32060 C9K8MH 129840818 Ki = 2300 nM T32060 C36AFR 129840841 Ki = 2500 nM T32060 CUD71X 129840856 Ki = 46 nM T32060 CV4D2F 129840894 Ki = 2650 nM T32060 C40HCZ 129840904 Ki = 167 nM T32060 CY7DS0 129840906 Ki = 120 nM T32060 CJX83W 129840907 Ki > 10000 nM T32060 C4PU0E 129840972 Ki = 184 nM T32060 C6K4NX 129840994 Ki = 465 nM T32060 C6Y7FB 129841007 Ki = 520 nM T32060 CKA0L7 129841015 Ki = 4460 nM T32060 CK1G0Y 129841036 Ki = 9 nM T32060 CGUW90 129841059 Ki > 5000 nM T32060 CV8SI7 129841063 Ki = 1.7 nM T32060 C10VDB 130431277 Ki = 7 nM T32060 CI1NF8 130431279 Ki = 90.4 nM T32060 CS8O4E 130431287 Ki = 25 nM T32060 C85MOW 130431289 Ki = 620 nM T32060 C2OH7B 130431291 Ki = 2990 nM T32060 CEQ43Y 130431295 Ki = 6600 nM T32060 CK64GU 130431296 Ki = 336 nM T32060 CYW0X2 130431314 Ki = 21.3 nM T32060 CDN26V 130431316 Ki = 28.1 nM T32060 CL64UW 130431317 Ki = 3.2 nM T32060 C8HE2O 130431318 Ki = 188 nM T32060 CZ6S4T 130431319 Ki = 940 nM T32060 C8ZHI7 130431325 Ki = 2.41 nM T32060 CF5SW8 130431328 Ki = 7600 nM T32060 CN9RZ3 130431329 Ki = 1933 nM T32060 CN70MW 130431337 Ki = 5.22 nM T32060 C4GF1U 130431342 Ki = 42.9 nM T32060 C2WI5R 130431351 Ki = 60.1 nM T32060 C50GOC 130442480 Ki = 8700 nM T32060 CM04RF 130442572 Ki = 4300 nM T32060 C5XZN0 132007291 Ki > 10000 nM T32060 CY8B9L 132060743 Ki = 1023 nM T32060 CGHO19 132060770 Ki = 475 nM T32060 CT81OY 132060776 Ki = 296 nM T32060 C7I5CQ 132118109 EC50 = 1600 nM T32060 CHB6K5 132118110 EC50 = 1860 nM T32060 CU8D9A 132118356 EC50 > 10000 nM T32060 C7KYG2 132118671 EC50 = 4950 nM T32060 CQX7N3 132118712 EC50 > 10000 nM T32060 C4LJ2Y 132503215 Ki = 286 nM T32060 CM8B1L 132525569 Ki = 12 nM T32060 CU5L0K 132525570 Ki = 10 nM T32060 CAVB41 132584404 Ki > 10000 nM T32060 CS0MB3 132938109 Ki = 2115 nM T32060 C8O2EP 134130246 Ki = 2041.74 nM T32060 CQX4U3 134133064 Ki > 10000 nM T32060 CCPI30 134133464 Ki = 0.38 nM T32060 C0J2ML 134133604 Ki = 748 nM T32060 CM0TS6 134133967 Ki = 251.19 nM T32060 CP3J9C 134134314 Ki = 1995.26 nM T32060 CZ8HL0 134134668 Ki > 10000 nM T32060 CR4F6X 134135492 Ki = 1.1 nM T32060 CM34TY 134135507 Ki = 0.24 nM T32060 C6G4CW 134135745 Ki > 10000 nM T32060 CGX03A 134136246 Ki = 1862.09 nM T32060 CD41CW 134137432 Ki = 1.2 nM T32060 C9A6KG 134138183 Ki > 10000 nM T32060 CH0FX4 134138769 Ki > 10000 nM T32060 C90XZH 134138881 Ki = 0.32 nM T32060 CTP83K 134139510 Ki = 0.34 nM T32060 CR7C9U 134139964 Ki = 1.585 nM T32060 CNSB82 134141050 Ki > 10000 nM T32060 CLW86T 134141354 Ki = 120 nM T32060 C68AXD 134141831 Ki > 10000 nM T32060 CXC80B 134142146 Ki = 3.3 nM T32060 CCS9A1 134142903 Ki = 7.943 nM T32060 CJFV62 134143302 Ki > 10000 nM T32060 C08RJA 134143536 Ki > 10000 nM T32060 C5L9BD 134143752 Ki > 10000 nM T32060 CVJ70S 134143778 Ki = 0.35 nM T32060 CV8IR0 134143977 Ki = 0.631 nM T32060 CR5L4K 134144303 Ki = 281 nM T32060 C71PIY 134144970 Ki > 10000 nM T32060 C8AZ1F 134146083 Ki = 4.3 nM T32060 C8RI0E 134146106 Ki = 2.2 nM T32060 CC9P2T 134146194 Ki = 1144 nM T32060 C19LRO 134146585 Ki > 10000 nM T32060 CUQ0F6 134147456 Ki = 6.31 nM T32060 C7S5RQ 134149008 Ki > 10000 nM T32060 CBU81N 134149168 Ki > 10000 nM T32060 COUJ52 134149355 Ki = 1.585 nM T32060 CAO9T6 134150123 Ki > 10000 nM T32060 CLU34D 134151427 Ki = 391.3 nM T32060 CK23XB 134151891 Ki = 0.87 nM T32060 C8PT9W 134152052 Ki > 10000 nM T32060 C73ISY 134152157 Ki > 10000 nM T32060 CI0G7H 134153418 Ki = 1.8 nM T32060 CB6M5Y 134153538 Ki = 483 nM T32060 CP41RT 134154065 Ki > 10000 nM T32060 C79TEI 134154068 Ki = 630.96 nM T32060 C9DQ4Y 134154208 Ki = 0.5 nM T32060 CMJ1U3 134154387 Ki = 975 nM T32060 C4VGJ5 134154679 Ki = 630.96 nM T32060 CU6C4G 134154943 Ki = 16 nM T32060 C6QAY2 134155116 Ki = 1202.26 nM T32060 C79QLN 134155460 Ki > 10000 nM T32060 CZFB29 134155462 Ki > 10000 nM T32060 CZJ15H 134155852 Ki = 25.12 nM T32060 CVR87Q 134156222 Ki = 1022 nM T32060 C7UOJ8 134156506 Ki > 10000 nM T32060 C5UQW2 134157367 Ki > 10000 nM T32060 C3BDA6 134157788 Ki > 10000 nM T32060 CF7EV5 134265590 EC50 = 100000 nM T32060 CR06XB 134265618 EC50 = 2510 nM T32060 CNA08H 134265620 EC50 = 53.2 nM T32060 C46YNU 134265622 EC50 = 1310 nM T32060 CA5PX2 134265627 EC50 = 37.2 nM T32060 CAS9Z4 134265663 EC50 = 236 nM T32060 CVY5G8 134265675 EC50 = 99.9 nM T32060 C6SLE4 134265705 EC50 = 100000 nM T32060 C8WAR6 134265732 EC50 = 980 nM T32060 C1GY2T 135156251 EC50 > 10000 nM T32060 C6N8GM 135367405 Ki = 159 nM T32060 C6LU0C 135367816 Ki = 399 nM T32060 CD2TH9 135367820 Ki = 471 nM T32060 C5AMD9 135367857 Ki = 138 nM T32060 C9ZCL5 135458672 Ki = 32700 nM T32060 C7AGR0 135474338 Ki > 100000 nM T32060 C0H9YX 135507495 Ki = 0.3981 nM T32060 CNI90F 135797785 Ki = 0.19 nM T32060 CE40DG 135882460 Ki = 2500 nM T32060 CG7LZ8 136020081 Ki = 352 nM T32060 C6G9TB 136020082 Ki = 284 nM T32060 C1VNH5 136020088 Ki > 1000 nM T32060 C2NWA6 136020089 Ki = 994 nM T32060 CUKO20 136020617 Ki > 10000 nM T32060 COF0U5 136020618 Ki > 10 nM T32060 CF89JI 136030596 Ki > 10000 nM T32060 CE8GB9 136030693 Ki > 10000 nM T32060 C65VFI 136030744 Ki > 10000 nM T32060 COIX80 136054961 Ki > 10000 nM T32060 C89VLZ 136056636 Ki = 7.9 nM T32060 CUG28I 136117980 Ki = 3.6 nM T32060 CB12QP 136152964 Ki = 491 nM T32060 CAE39V 136188797 Ki > 10000 nM T32060 CLAP52 136259032 Ki > 10000 nM T32060 C9EIP8 137631570 IC50 = 651 nM T32060 CBX2V5 137631812 EC50 > 10000 nM T32060 CHM36P 137631892 Ki = 336 nM T32060 CQO58W 137632042 EC50 > 10000 nM T32060 CDQ6X3 137632069 EC50 = 93 nM T32060 CS5K0I 137632108 EC50 = 3700 nM T32060 C64KPN 137632218 EC50 > 10000 nM T32060 C96DFN 137632449 EC50 = 238 nM T32060 CN8BJ2 137632607 Ki = 3700 nM T32060 C3R2LO 137632761 Ki = 5400 nM T32060 CMO30D 137633009 EC50 > 10000 nM T32060 C3PF9Z 137633454 Ki = 1500 nM T32060 COF9I6 137633705 Ki = 2.6 nM T32060 CU01TV 137633827 Ki > 10000 nM T32060 C8YM6U 137633863 Ki = 100 nM T32060 C5ZL0C 137633983 EC50 > 10000 nM T32060 CN1I7A 137634153 Ki = 3600 nM T32060 CATU84 137634233 EC50 > 10000 nM T32060 C6FRJ5 137634397 Ki = 880 nM T32060 CXCJ60 137634432 EC50 > 10000 nM T32060 C9M3RV 137635151 EC50 = 457.09 nM T32060 C94MFJ 137635172 EC50 > 10000 nM T32060 CC51JN 137635185 Ki = 1703 nM T32060 CNR82A 137635294 IC50 = 17 nM T32060 CPHI76 137635364 Ki = 520 nM T32060 C6DH9X 137635433 IC50 = 3.4 nM T32060 C8ZFQ6 137635685 Ki = 200 nM T32060 C5N4PR 137635711 EC50 > 10000 nM T32060 C0K3AP 137635725 IC50 = 25 nM T32060 CJT0A2 137635932 EC50 > 10000 nM T32060 C05XCQ 137635978 Ki = 2.692 nM T32060 CBH98Q 137635994 EC50 = 4260 nM T32060 CZ36LE 137636066 Ki = 2000 nM T32060 CAL1W4 137636298 Ki > 20000 nM T32060 CAQ6I5 137636351 Ki = 6.3 nM T32060 CFM92C 137636384 Ki = 65 nM T32060 CPQ34V 137636430 EC50 > 10000 nM T32060 CQ71WO 137636435 EC50 > 10000 nM T32060 C6GWQ3 137636460 Ki = 310 nM T32060 C8Z1XW 137636480 EC50 = 27.54 nM T32060 CQ20FO 137636498 Ki = 39 nM T32060 CZU6N5 137636581 Ki > 10000 nM T32060 C4OT7C 137637069 EC50 > 5000 nM T32060 CTD64R 137637165 EC50 > 10000 nM T32060 C0YDQ5 137637428 Ki = 2100 nM T32060 CK29VL 137637650 EC50 > 10000 nM T32060 C71BUE 137637880 EC50 = 721 nM T32060 CDX39B 137637994 Ki = 691 nM T32060 C56GTL 137638508 EC50 > 10000 nM T32060 CM0DJ5 137638903 EC50 > 10000 nM T32060 C49VDK 137638973 Ki = 880 nM T32060 C1HX3Z 137639304 Ki > 20000 nM T32060 CK8UC2 137639485 EC50 > 10000 nM T32060 CEQ68W 137639630 EC50 > 10000 nM T32060 CPQ83I 137639705 EC50 > 10000 nM T32060 C5KX6V 137640062 EC50 = 138.04 nM T32060 CC16HE 137640152 Ki = 4200 nM T32060 CZP68A 137640189 Ki = 430 nM T32060 CB2NO0 137640203 Ki = 78 nM T32060 CKJD12 137640272 EC50 = 144.54 nM T32060 CV49MZ 137640371 Ki = 2300 nM T32060 CCU7L3 137640391 Ki = 380 nM T32060 C3U5NF 137640522 IC50 = 89 nM T32060 CPK8A0 137640608 EC50 = 1862.09 nM T32060 C8IO0R 137640836 Ki = 2800 nM T32060 C62QAM 137640945 EC50 = 2220 nM T32060 CWQ80N 137640967 IC50 = 37.6 nM T32060 C90GKM 137641125 EC50 > 10000 nM T32060 CUQ8F5 137641376 EC50 > 10000 nM T32060 C3LYX9 137641832 Ki > 10000 nM T32060 C4I6QS 137641944 IC50 = 21.46 nM T32060 C6PT7L 137642033 Ki > 20000 nM T32060 C5WS6Q 137642134 Ki = 156 nM T32060 C6P9FW 137642149 EC50 > 10000 nM T32060 C94WSH 137642380 Ki = 4.9 nM T32060 C4HJ1N 137642593 EC50 = 463 nM T32060 CO6J9Q 137642857 EC50 > 10000 nM T32060 CAC6W0 137643122 Ki = 600 nM T32060 C71XIQ 137643132 Ki = 2700 nM T32060 CK51LB 137643309 Ki = 2200 nM T32060 CMJU75 137643395 IC50 = 26.4 nM T32060 CX65BH 137643424 EC50 = 655 nM T32060 CPL0K5 137643658 EC50 > 10000 nM T32060 C1ZP9R 137643846 EC50 = 398 nM T32060 C3O0FX 137643951 Ki = 300 nM T32060 CK5HG6 137644041 Ki = 5.754 nM T32060 CIKD85 137644487 EC50 > 10000 nM T32060 CWUM83 137644521 Ki > 10000 nM T32060 CDA80E 137644790 Ki = 179 nM T32060 C34PUI 137644833 Ki = 180 nM T32060 CRGN16 137644935 EC50 = 1090 nM T32060 CVX6T1 137644966 Ki = 5.6 nM T32060 CSO38A 137645024 EC50 > 5000 nM T32060 C4PV8U 137645196 Ki = 6400 nM T32060 CHT42S 137645295 IC50 = 9.5 nM T32060 CZ8CU6 137645501 Ki = 530 nM T32060 CNH95X 137645574 Ki = 2200 nM T32060 CRU20V 137645667 EC50 > 10000 nM T32060 CA7P4F 137645674 EC50 > 10000 nM T32060 C3TP2G 137645830 Ki = 480 nM T32060 CUR7T5 137645858 EC50 > 10000 nM T32060 CCP38D 137645926 Ki = 152 nM T32060 CVX74E 137646045 Ki = 489 nM T32060 C5Q6DL 137646111 EC50 > 10000 nM T32060 CPI68E 137646281 Ki = 1415 nM T32060 C8PV0N 137646568 IC50 = 6.4 nM T32060 C4YE8H 137646603 EC50 = 436.52 nM T32060 C9EYB1 137646716 EC50 > 10000 nM T32060 C2O1XW 137646874 EC50 > 10000 nM T32060 C6C3IK 137646921 EC50 > 10000 nM T32060 CN5R7Q 137647004 EC50 > 10000 nM T32060 CD2TE0 137647007 EC50 > 10000 nM T32060 C5Y0FG 137647246 EC50 > 10000 nM T32060 CU6V5W 137647439 EC50 = 269.15 nM T32060 CYH5U9 137647533 Ki = 2300 nM T32060 CA48GB 137647635 EC50 = 635 nM T32060 CO5U9A 137647674 IC50 = 1160 nM T32060 CQA0B2 137647926 EC50 = 884 nM T32060 CR64OK 137648428 EC50 = 2951.21 nM T32060 C4HX6J 137648810 EC50 > 10000 nM T32060 C2VBA0 137649655 EC50 = 2511.89 nM T32060 CMXI62 137649997 Ki = 646 nM T32060 CB4HG5 137650482 IC50 = 331 nM T32060 CWQF69 137650550 IC50 = 5.12 nM T32060 C52IRM 137650705 Ki = 197 nM T32060 C1GZV3 137650863 EC50 = 307 nM T32060 CKG08R 137650961 Ki = 665 nM T32060 CR3Z6M 137651073 Ki = 410 nM T32060 CXV3D7 137651249 EC50 > 10000 nM T32060 CW4T6D 137651322 Ki = 2900 nM T32060 C47TWK 137651544 IC50 = 34.4 nM T32060 C1SY4J 137651715 EC50 >= 1800 nM T32060 C15YDU 137651936 Ki = 1200 nM T32060 CVK26R 137652044 Ki = 410 nM T32060 C51CGJ 137652310 Ki = 139 nM T32060 CTE69H 137652480 EC50 = 75 nM T32060 CY59NZ 137652713 EC50 > 10000 nM T32060 CX30HQ 137653096 Ki > 20000 nM T32060 CPFG35 137653140 EC50 = 674 nM T32060 C04XYN 137653567 IC50 = 9.14 nM T32060 CC12VB 137653689 EC50 > 10000 nM T32060 C2E3FV 137653850 Ki = 157 nM T32060 C4C6EV 137653986 Ki > 20000 nM T32060 CKT1F5 137654351 EC50 > 10000 nM T32060 COTX19 137654511 Ki > 20000 nM T32060 C6N0DT 137654586 IC50 = 7.1 nM T32060 CF5Y2A 137654675 Ki = 3600 nM T32060 CS1Y8F 137654798 EC50 > 10000 nM T32060 C0SKV1 137654850 Ki > 10000 nM T32060 CZ50SL 137654926 EC50 > 10000 nM T32060 CLI4D8 137655029 Ki = 1000 nM T32060 CJMR75 137655187 EC50 = 1310 nM T32060 C53QIZ 137655324 EC50 = 23.99 nM T32060 C4VG0U 137655411 Ki = 371 nM T32060 C7RW9H 137655451 Ki = 1600 nM T32060 CHI8M2 137655535 EC50 > 10000 nM T32060 CJAZ13 137655556 Ki = 9000 nM T32060 C6CA5H 137655594 Ki > 20000 nM T32060 CB20MW 137655657 EC50 = 1288.25 nM T32060 C91UBP 137655705 EC50 > 10000 nM T32060 CDAN02 137655735 Ki = 120 nM T32060 C1PKE6 137655741 EC50 > 10000 nM T32060 CD16SQ 137655795 Ki = 160 nM T32060 CKW87Y 137655846 EC50 > 10000 nM T32060 CZ82HF 137655858 EC50 = 6760.83 nM T32060 C60XIF 137655882 EC50 > 10000 nM T32060 CXH16S 137655884 Ki = 75.8 nM T32060 C17NVY 137656030 EC50 > 10000 nM T32060 CVEN03 137656381 IC50 = 2300 nM T32060 CL8RT7 137656524 EC50 > 10000 nM T32060 C1SX4C 137656726 EC50 = 77 nM T32060 CA7F5N 137657115 Ki = 94 nM T32060 CV2CR4 137657153 Ki = 1100 nM T32060 CCKP95 137657310 EC50 = 147.91 nM T32060 CE0Y7P 137657322 Ki > 15000 nM T32060 CRT86S 137657427 Ki = 3400 nM T32060 CME6U8 137657882 Ki = 562.34 nM T32060 CEJ9L8 137657949 IC50 = 71.3 nM T32060 CH76FP 137657951 Ki > 20000 nM T32060 CKQ7Y9 137658074 EC50 > 10000 nM T32060 C0OI2B 137658246 EC50 > 10000 nM T32060 C3LHT5 137658253 IC50 = 44 nM T32060 CH9R5V 137658409 EC50 > 5000 nM T32060 CBK37P 137658537 EC50 = 3530 nM T32060 C8G0HO 137658832 IC50 = 244 nM T32060 CFQ7C9 137659145 IC50 = 60 nM T32060 C3JG5Z 137659281 EC50 > 10000 nM T32060 CEZ07P 137659303 Ki = 250 nM T32060 CLQX32 137659728 IC50 = 2.87 nM T32060 CP9AN6 137659990 Ki = 1600 nM T32060 CP6US4 137660046 Ki = 1300 nM T32060 CAM68B 137660072 EC50 > 5000 nM T32060 C5Q9CM 137660307 EC50 = 70.79 nM T32060 CF9RZ5 137660385 IC50 = 26.2 nM T32060 C3UHP5 137660422 EC50 > 10000 nM T32060 C5V4DQ 137660707 Ki > 20000 nM T32060 CX4D7Y 137660741 Ki = 161 nM T32060 C42IDE 137660837 Ki = 2000 nM T32060 C6SHF4 137661018 EC50 > 10000 nM T32060 CO2TV7 137661051 EC50 = 1862.09 nM T32060 C0YZF2 137661221 EC50 > 5000 nM T32060 CEJ38Q 137661378 EC50 = 281.84 nM T32060 C8JH6R 137661673 EC50 = 151 nM T32060 CN52AG 137662193 EC50 > 10000 nM T32060 C0R6XM 138691314 Ki > 10000 nM T32060 CU3Y7W 138691316 Ki > 10000 nM T32060 CH2W4P 138691317 Ki > 10000 nM T32060 CHSC40 138691321 Ki = 8511 nM T32060 C18UZA 138691329 Ki > 10000 nM T32060 C1XWV0 138691338 Ki > 10000 nM T32060 C6LE1A 138691362 Ki > 10000 nM T32060 CN9R4A 138691364 Ki > 10000 nM T32060 C8H2KR 138691366 Ki > 10000 nM T32060 CJ43GI 139187858 Ki > 10000 nM T32060 C47QCK 139187859 Ki = 55 nM T32060 C2Z9CD 139488518 Ki > 10000 nM T32060 CJK95T 139488527 Ki > 10000 nM T32060 CAF2H8 139488606 Ki > 10000 nM T32060 C54CIL 139488740 Ki > 10000 nM T32060 COT18S 145011254 Ki > 10000 nM T32060 CLJW61 145955880 Ki = 42 nM T32060 CMO17A 145960744 Ki = 27 nM T32060 CAJ7P6 145961144 Ki = 75 nM T32060 C67GQI 145961372 Ki = 2608 nM T32060 C59KNW 145961441 Ki = 30 nM T32060 CI4H8B 145961535 Ki = 155 nM T32060 C8PTZ7 145961730 Ki = 47 nM T32060 CQ4RA7 145961842 Ki = 8 nM T32060 C1YE4Q 145962266 Ki = 91 nM T32060 C71HNB 145962633 Ki > 10000 nM T32060 C9G5YC 145962760 Ki > 5000 nM T32060 C56BKQ 145962801 Ki = 1158 nM T32060 CVM9G4 145962946 Ki = 9.5 nM T32060 CFA09Q 145962985 Ki = 2434 nM T32060 CO7P1B 145963059 Ki > 5000 nM T32060 C85BSY 145963127 Ki = 793 nM T32060 C9B0SZ 145963169 Ki = 56 nM T32060 C2ZSA4 145963224 Ki = 30 nM T32060 CDTR93 145963270 Ki = 138 nM T32060 CNA8I5 145963810 Ki = 22 nM T32060 C7KC3T 145963830 Ki = 1100 nM T32060 CEN94V 145963961 IC50 = 113 nM T32060 C3I6YP 145963975 IC50 = 83.2 nM T32060 C4Y2AL 145964000 Ki > 5000 nM T32060 CE32PV 145964143 Ki = 46.8 nM T32060 CHDN35 145964150 Ki = 2200 nM T32060 C1KH2E 145964159 Ki = 1400 nM T32060 C1B8QW 145964299 IC50 = 247 nM T32060 C95NZO 145964427 Ki = 159 nM T32060 C0N8KC 145964622 IC50 = 167 nM T32060 C6T4RY 145964846 Ki = 76 nM T32060 C24NSP 145964857 Ki = 12.5 nM T32060 C7MBS0 145964982 IC50 = 53.9 nM T32060 C12OVL 145965034 Ki > 10000 nM T32060 C7JS9I 145965041 IC50 = 1280 nM T32060 C9D8IB 145965203 Ki = 527 nM T32060 CA8KF0 145965309 Ki > 5000 nM T32060 C5DL3N 145965355 Ki = 102 nM T32060 CV07EO 145965433 IC50 = 67.5 nM T32060 C9KXP6 145965474 Ki = 408 nM T32060 CKO51D 145965628 Ki = 240 nM T32060 CLP94W 145965668 Ki = 452 nM T32060 C8TF9G 145965840 Ki = 343 nM T32060 C5W4LM 145965940 Ki > 10000 nM T32060 C4EQ9C 145966293 EC50 = 2880 nM T32060 CLM10C 145966333 IC50 = 154 nM T32060 C1T4DN 145966418 Ki = 351 nM T32060 CRS7V6 145966748 Ki = 400 nM T32060 C5L4WF 145967359 IC50 = 95.5 nM T32060 C81VUO 145967771 Ki > 10 nM T32060 CJS56K 145967795 Ki > 10000 nM T32060 CG4A3U 145968880 IC50 = 29.5 nM T32060 CM6HG9 145968927 IC50 = 523 nM T32060 CB01DY 145969032 IC50 = 39.8 nM T32060 C2A0FO 145969167 IC50 = 94.2 nM T32060 CR5ZQ6 145969279 IC50 = 56.23 nM T32060 CQ8EM6 145969402 Ki = 68 nM T32060 CI5R8W 145969406 Ki = 7 nM T32060 CE3WK8 145969738 IC50 = 36.31 nM T32060 CZ9HC2 145970712 IC50 = 46.7 nM T32060 CT2LQ4 145970743 Ki = 20 nM T32060 CQC6Y1 145970782 Ki = 56 nM T32060 CRC9T0 145971556 IC50 = 476 nM T32060 C8A2XG 145971561 Ki = 270 nM T32060 CB43OV 145971604 Ki = 6 nM T32060 CQJ5O8 145971635 Ki = 6900 nM T32060 C56RAO 145972025 Ki = 404 nM T32060 C7BVC1 145972374 Ki = 310 nM T32060 CR06QO 145972382 IC50 = 89.9 nM T32060 CWRM23 145972513 IC50 = 42.2 nM T32060 C79TNE 145972796 Ki > 10000 nM T32060 C1QY4E 145973003 Ki = 8 nM T32060 CEOY46 145973577 Ki = 220 nM T32060 CT51VH 145974031 Ki = 20 nM T32060 C6XIN0 145974114 Ki > 10000 nM T32060 C6AGN3 145974143 IC50 = 52.4 nM T32060 CW6EX3 145974189 Ki = 1352 nM T32060 C9L7EM 145974368 Ki = 6.5 nM T32060 CD8ZL6 145974750 Ki > 10 nM T32060 CDOJ39 145974939 IC50 = 64.9 nM T32060 CR83MU 145975214 IC50 = 910 nM T32060 CJF4Z0 145975393 IC50 = 134 nM T32060 CZ39GQ 145975595 IC50 = 62.4 nM T32060 COY2P3 145975720 Ki = 59 nM T32060 CL7EX5 145975776 Ki = 2805 nM T32060 C7R2MD 145975905 Ki = 496 nM T32060 C71CYU 145975946 Ki = 3900 nM T32060 C0V4AL 145975992 Ki = 259 nM T32060 C2TN8W 145976085 Ki = 5800 nM T32060 C8XFM7 145976120 Ki = 772 nM T32060 CB2R6J 145976187 Ki = 10 nM T32060 CCDU50 145976348 IC50 = 152 nM T32060 CZ5XK2 145976408 Ki = 715 nM T32060 C34XME 145976696 Ki = 245 nM T32060 C9FR7N 145976732 IC50 = 106 nM T32060 CNCS36 145976746 Ki = 58 nM T32060 C7L9DG 145976983 Ki = 310 nM T32060 CXDR94 145977222 Ki = 498 nM T32060 C8NW7Y 145977256 Ki = 75 nM T32060 C6BFY7 145977338 Ki > 10000 nM T32060 C8DP4I 145977442 Ki = 48.7 nM T32060 C3BI1R 145978113 Ki > 10000 nM T32060 C72SMR 145978208 IC50 = 324 nM T32060 C8VL3Y 145978472 Ki = 17330 nM T32060 CQU8R0 145978665 Ki > 10000 nM T32060 C6AV9G 145978819 Ki > 10000 nM T32060 C1Q2BR 145978965 IC50 = 81.5 nM T32060 C2PK6X 145980101 Ki = 64 nM T32060 C87MSW 145980271 Ki = 6059 nM T32060 CD92WV 145980513 Ki > 10000 nM T32060 C8I7QL 145980875 Ki = 889 nM T32060 C6H7SC 145981004 Ki = 48 nM T32060 CC2UQ5 145981118 Ki = 4565 nM T32060 C4AF0G 145981310 IC50 = 314 nM T32060 C67AIW 145981408 IC50 = 32 nM T32060 C7LBY5 145982138 Ki = 42 nM T32060 CO7WP6 145982353 IC50 = 84.9 nM T32060 CEK60A 145982506 Ki = 244 nM T32060 CI59TX 145983018 Ki = 2453 nM T32060 CYC58R 145983059 Ki = 7 nM T32060 C4F5OT 145983128 Ki = 451 nM T32060 C5ZG9M 145983139 Ki = 49 nM T32060 CV2GU9 145983144 Ki = 1400 nM T32060 C4PKM2 145983390 Ki = 26 nM T32060 CIAF74 145983468 Ki = 30 nM T32060 CE7MF4 145983751 Ki = 35 nM T32060 CDQ4U7 145983760 Ki = 51 nM T32060 CYW9B2 145983794 Ki = 64 nM T32060 C1DW4U 145983928 IC50 = 24.6 nM T32060 C8I1WG 145983961 Ki = 10 nM T32060 CP5H4D 145984065 Ki = 1904 nM T32060 C58DHN 145984151 IC50 = 254 nM T32060 CJ35DM 145984299 Ki = 13 nM T32060 CU7E4M 145984511 Ki = 24 nM T32060 C6JUY0 145984737 Ki = 18 nM T32060 CID02G 145984807 Ki = 2040 nM T32060 CP9D3A 145984902 Ki = 28 nM T32060 CM5X3V 145985050 Ki = 6 nM T32060 CG10LK 145985224 Ki = 30 nM T32060 CFJ9B3 145985233 Ki = 12 nM T32060 C5AOI6 145985289 Ki = 29 nM T32060 CW30NA 145985505 Ki = 41 nM T32060 C7ZRP1 145985527 Ki = 1150 nM T32060 C2XY8Q 145985533 Ki = 16 nM T32060 C7NI4X 145985585 Ki = 33 nM T32060 C9LJ5T 145985692 Ki = 15 nM T32060 C7QIX0 145985718 Ki = 29 nM T32060 C6V5QS 145985823 Ki = 5 nM T32060 C07GKD 145985958 Ki = 1970 nM T32060 CCM18E 145986031 Ki = 35 nM T32060 CR0XQ3 145986138 Ki = 16 nM T32060 CXC79K 145986552 IC50 = 7250 nM T32060 CNJH37 145986752 Ki = 900 nM T32060 CZ5O8R 145987659 IC50 = 113 nM T32060 COS58J 145987942 IC50 = 82.3 nM T32060 C6MHU2 145988006 IC50 = 546 nM T32060 C9ZBE8 145988017 Ki = 200 nM T32060 CHOB70 145988038 IC50 = 134 nM T32060 C86XQR 145988313 Ki = 2460 nM T32060 C9W1QA 145988497 IC50 = 1.1 nM T32060 CUGO10 145988693 Ki = 164 nM T32060 CVC14L 145989181 IC50 = 130 nM T32060 CR2EV8 145989183 IC50 = 1660 nM T32060 C39CSX 145989329 Ki > 10000 nM T32060 CMJL94 145989451 IC50 = 2840 nM T32060 C41SBL 145990126 IC50 = 34 nM T32060 CK5IA4 145990443 Ki = 106 nM T32060 CE9PT1 145990482 IC50 = 956 nM T32060 CKWF21 145990750 Ki > 10000 nM T32060 CMJ46R 145990794 IC50 = 27.5 nM T32060 C5TNP0 145991127 IC50 = 318 nM T32060 CW14AE 145991244 IC50 = 10.4 nM T32060 C7RJ4E 145991363 Ki = 3000 nM T32060 CU6E1Z 145991746 IC50 = 82.4 nM T32060 CI1EQ3 145991900 Ki = 286 nM T32060 C9WME0 145992265 Ki = 66 nM T32060 C5DVK4 145992403 Ki = 1595 nM T32060 CCP2U1 145992489 Ki = 1105 nM T32060 CELG57 145992523 IC50 = 282 nM T32060 CB64KH 145992860 IC50 = 854 nM T32060 C9PS8N 145993117 IC50 = 25.9 nM T32060 CT63XO 145993172 IC50 = 0.6 nM T32060 C0Z6YX 145993493 IC50 = 29.1 nM T32060 CQ93KE 145993540 Ki = 1.92 nM T32060 C17HSV 145993577 IC50 = 103 nM T32060 CX1N0L 145993740 Ki > 5000 nM T32060 CO1BX3 145994087 Ki = 70 nM T32060 CS1LF2 145994186 Ki = 4 nM T32060 CC2G1V 146025727 Ki = 3400 nM T32060 C5ZOJ3 146680920 Ki = 3355 nM T32060 CV9G7Z 153287572 Ki > 10000 nM T32060 CO85KL 153287574 Ki > 10000 nM T32060 CZ1K4D 155510674 Ki = 205 nM T32060 CC3KP7 155510927 Ki = 794 nM T32060 CM4RB0 155511262 Ki = 29 nM T32060 C9KX6O 155511928 Ki = 147 nM T32060 CU4H6L 155512064 Ki = 2313 nM T32060 CXF90M 155512487 Ki = 11 nM T32060 CO68LC 155512944 Ki > 10000 nM T32060 C90FST 155513438 Ki = 22 nM T32060 C95QOT 155514378 Ki = 1552 nM T32060 CK9YN0 155514430 Ki = 470 nM T32060 CI4DT8 155514575 Ki = 891 nM T32060 CJUI87 155514774 Ki = 23 nM T32060 C4X2RG 155515318 Ki = 33 nM T32060 C3NB0D 155515324 Ki = 11590 nM T32060 C0Q8PR 155515407 Ki = 1490 nM T32060 CWO56B 155515415 Ki > 10000 nM T32060 C2TN5D 155515890 Ki = 892 nM T32060 C7KT0D 155515919 Ki = 1660 nM T32060 C13LOV 155515942 Ki = 1412 nM T32060 CUM2N4 155515982 Ki = 65 nM T32060 C7OF4C 155516118 Ki = 32 nM T32060 CG5M1O 155516282 Ki = 1927 nM T32060 CEA9D5 155517238 Ki = 1888 nM T32060 CW0B5K 155518159 Ki > 10000 nM T32060 CYB12O 155518974 Ki = 60100 nM T32060 CCEZ93 155519102 Ki = 1830 nM T32060 CQD2J7 155519393 Ki = 843 nM T32060 C2SXT1 155519515 Ki = 596 nM T32060 C0KLD8 155519559 Ki = 1003 nM T32060 C07BTO 155519598 Ki = 773 nM T32060 C5FL7R 155520499 Ki = 533 nM T32060 C8OC3W 155520552 Ki = 177 nM T32060 CQ76MP 155521503 Ki = 1047 nM T32060 C1OS6D 155522116 Ki = 2291 nM T32060 C98RDQ 155522218 Ki = 433 nM T32060 C2TV4Y 155522487 Ki > 10000 nM T32060 CP6H1D 155522562 Ki = 322 nM T32060 CUG8L3 155522920 Ki > 10000 nM T32060 CUG4Q8 155523121 Ki = 1230 nM T32060 CD9QU6 155523519 Ki = 91 nM T32060 C2Y9CW 155523745 Ki = 2099 nM T32060 C5KYB4 155524228 Ki = 209 nM T32060 CK4B0R 155524491 Ki = 609 nM T32060 CUO93F 155524808 Ki = 342 nM T32060 CQB0M8 155524884 Ki > 10000 nM T32060 C65UZD 155524956 Ki = 548 nM T32060 CGS21U 155525549 Ki > 10000 nM T32060 CZ81JA 155526026 Ki = 266 nM T32060 C1U2XO 155526651 Ki = 222 nM T32060 CRF1A0 155527638 EC50 = 45.71 nM T32060 CW68KC 155528355 Ki > 10000 nM T32060 C7C1EF 155528967 Ki = 435 nM T32060 C5J7AU 155529153 Ki = 376 nM T32060 C9KS5C 155529450 Ki = 167 nM T32060 CEN90X 155529453 Ki = 358 nM T32060 CKZ25Y 155529679 Ki = 922 nM T32060 C7UZI1 155530285 Ki = 3236 nM T32060 C3X4IA 155530328 Ki = 361 nM T32060 C9PC3D 155530350 Ki = 1526 nM T32060 CVLC03 155530779 Ki = 216 nM T32060 C98YQF 155531012 Ki = 283 nM T32060 C4W6VC 155531065 Ki = 175 nM T32060 CV6ST2 155531084 Ki = 434 nM T32060 C5HWP4 155531362 Ki > 10000 nM T32060 CCT8V9 155531846 Ki = 2628 nM T32060 CX43DV 155532107 EC50 = 2.692 nM T32060 C5XNT1 155532396 Ki = 2455 nM T32060 CX6DV4 155533028 Ki = 3983 nM T32060 C23GDV 155533534 Ki = 1277 nM T32060 CSY06A 155533573 Ki > 10000 nM T32060 C3OEH2 155533648 Ki = 1918 nM T32060 C15RYP 155533660 Ki > 10000 nM T32060 CZA89B 155533824 Ki = 3.22 nM T32060 CY01GZ 155533850 Ki = 1488 nM T32060 CP3J8B 155534152 Ki = 107 nM T32060 C3L0CP 155534184 Ki = 325 nM T32060 CG85SB 155534301 Ki = 43 nM T32060 C3VGT0 155534362 Ki = 21 nM T32060 C3JPS4 155534559 EC50 = 122 nM T32060 CW7SV9 155534575 Ki = 183 nM T32060 C75FSY 155534794 Ki = 490 nM T32060 C6KAU3 155534798 Ki = 2020 nM T32060 C6KF4E 155535154 Ki = 1191 nM T32060 CGZ5T8 155535272 Ki = 53 nM T32060 C14JEX 155535878 Ki = 1175 nM T32060 C7OIP3 155535969 EC50 = 1819.7 nM T32060 CB79ZW 155536080 Ki > 10000 nM T32060 C5I1JA 155536087 Ki = 307 nM T32060 C7FVE8 155537034 Ki > 10000 nM T32060 C36FRH 155537074 Ki = 131 nM T32060 CD75GP 155537227 Ki > 10000 nM T32060 CB8IC7 155538144 Ki > 10000 nM T32060 C5F2GI 155538236 Ki = 725 nM T32060 C9TIU2 155538367 Ki > 10000 nM T32060 CYC1P3 155538451 Ki = 461 nM T32060 CM08NT 155538716 Ki > 10000 nM T32060 CAT98F 155539483 Ki = 1944 nM T32060 C6S8BA 155539600 Ki = 407 nM T32060 C4FJL0 155539960 EC50 = 352 nM T32060 C42GUK 155540147 Ki = 8913 nM T32060 C72KHI 155540514 EC50 = 22.91 nM T32060 C1JM5R 155540523 Ki = 1138 nM T32060 C2OWD4 155540721 Ki = 7413 nM T32060 CR2K1T 155540795 Ki = 661 nM T32060 CNU92V 155540807 Ki = 31 nM T32060 COS2E7 155541072 Ki > 10000 nM T32060 CMP8Q2 155541547 Ki = 1905 nM T32060 C6SU1V 155541676 Ki > 10000 nM T32060 CP7UG2 155541866 Ki = 35 nM T32060 COZ46W 155541871 Ki = 429 nM T32060 CXCW81 155542321 Ki = 430 nM T32060 C9FS3Y 155542461 Ki > 10000 nM T32060 C18OPI 155542619 Ki = 173 nM T32060 CT6HY4 155543250 Ki = 9333 nM T32060 C68MSK 155543653 Ki = 590 nM T32060 CZ7O0A 155544139 Ki = 197 nM T32060 CGU5M0 155544723 Ki > 10000 nM T32060 CD84VK 155544810 Ki = 540 nM T32060 C2XZD8 155545087 Ki = 251 nM T32060 CO9X1Z 155545526 Ki > 10000 nM T32060 CI0YL8 155545625 Ki > 10000 nM T32060 C74GFO 155546189 Ki = 376 nM T32060 CH3W9N 155546350 Ki > 10000 nM T32060 CD02EN 155547436 Ki = 334 nM T32060 COJ27N 155547693 Ki = 2274 nM T32060 CAT9X4 155548275 Ki = 7943 nM T32060 CSX3M0 155548666 EC50 = 154.88 nM T32060 C5LYE8 155548677 Ki = 42 nM T32060 C87JGN 155549153 Ki > 10000 nM T32060 CGP8O5 155549315 Ki = 456 nM T32060 C52FRY 155549978 Ki = 321 nM T32060 C7KWB9 155550387 Ki = 450 nM T32060 C8HPN7 155551113 Ki = 524 nM T32060 CN39VC 155551164 EC50 = 30.9 nM T32060 C61IVC 155551353 Ki > 10000 nM T32060 CHS71N 155551685 Ki = 209 nM T32060 C6E9LK 155552054 Ki = 652 nM T32060 CX8JA1 155552185 Ki = 130 nM T32060 CA1WS9 155552212 Ki = 406 nM T32060 C0DQ3Z 155552695 Ki = 140 nM T32060 CDQ7C2 155552798 Ki = 4354 nM T32060 CPV35U 155552826 Ki > 10000 nM T32060 CKF75H 155554324 Ki = 423 nM T32060 C6ZSU3 155554462 Ki = 197 nM T32060 C0PBT3 155555147 Ki > 10000 nM T32060 C2E5TR 155555506 Ki = 199 nM T32060 CUNK28 155555525 Ki = 1122 nM T32060 CYP63A 155556311 Ki = 194 nM T32060 CO52HW 155556527 Ki = 1698 nM T32060 C1N5VF 155556756 Ki > 10000 nM T32060 C5QYS0 155557134 Ki = 578 nM T32060 CD2L3K 155557443 Ki > 10000 nM T32060 CER48T 155557500 Ki > 10000 nM T32060 C4AG0H 155558726 Ki = 4700 nM T32060 C5L8HB 155560629 EC50 = 38.02 nM T32060 COG70U 155560942 Ki = 676 nM T32060 C9LV7U 155561048 EC50 = 316.23 nM T32060 C2HF6P 155561581 Ki = 406 nM T32060 CSK27Q 155561712 Ki = 414 nM T32060 C5O8AU 155561865 Ki > 10000 nM T32060 COL7N8 155561901 Ki > 10000 nM T32060 CL45NV 155561914 Ki = 1766 nM T32060 CW7M1D 155561995 Ki = 484 nM T32060 C93KWN 155562202 Ki = 337 nM T32060 CO3C6L 155562423 Ki > 10000 nM T32060 C5AI0S 155562519 Ki = 118 nM T32060 C5BQ8U 155562652 Ki = 314 nM T32060 CF6B4W 155562834 Ki = 443 nM T32060 CZ6IA2 155562918 Ki = 17170 nM T32060 CRCW25 155562997 Ki = 50 nM T32060 CG1L8E 155563286 Ki > 10000 nM T32060 C38WXS 155563374 Ki = 2589 nM T32060 C0INS4 155563826 Ki = 5129 nM T32060 C8YPA7 155564299 EC50 = 162 nM T32060 CR12DI 155565189 Ki = 970 nM T32060 C2MIU5 155565813 Ki = 96 nM T32060 C7P5VG 155566191 Ki = 41 nM T32060 CU46EB 155566665 Ki > 10000 nM T32060 C67LAG 155566854 Ki = 100 nM T32060 CW1TN7 155566925 Ki > 10000 nM T32060 C41UWT 155567307 Ki = 717 nM T32060 C4EX7C 155568246 Ki = 499 nM T32060 CXP3E4 155568794 Ki = 28 nM T32060 CB5IP9 155569021 Ki = 493 nM T32060 CP9V7M 155569396 Ki > 10000 nM T32060 C3ZNX6 155569414 Ki = 1290 nM T32060 CZ8RV4 155569568 Ki = 607 nM T32060 CP9TR0 10324985 Ki = 41.5 nM T32060 C6ZSL7 136016497 Ki = 173 nM T32060 CE2J8F 136016507 Ki = 235 nM T32060 CKM28Y 136016513 Ki = 655 nM T32060 CB2VD8 44241743 Ki = 0.54 nM T32060 D00APD 15124 Ki = 7600 nM T32060 D00AVR 135476741 Ki = 598 nM T32060 D00BWZ 10823903 Ki > 10000 nM T32060 D00EMF 3644637 Ki = 158.49 nM T32060 D00GOY 6604042 Ki = 351 nM T32060 D00GSD 25107716 Ki = 626 nM T32060 D00LXH 10753358 Ki = 158.49 nM T32060 D00NQV 5041 Ki = 273 nM T32060 D00NST 44452811 Ki = 0.78 nM T32060 D00OBS 44559159 Ki > 10000 nM T32060 D00OCV 44404892 Ki = 122 nM T32060 D00WEQ 62065 Ki = 0.6 nM T32060 D00YEB 25141414 Ki = 56 nM T32060 D00YVE 10219723 EC50 = 466 nM T32060 D01BGW 11708275 Ki = 16 nM T32060 D01CGM 3033677 Ki = 0.13 nM T32060 D01CXD 10398175 Ki = 20 nM T32060 D01HJZ 83632 Ki = 7356 nM T32060 D01HRV 9847194 IC50 = 1100 nM T32060 D01JXM 46222048 Ki > 1000 nM T32060 D01KAX 135453290 Ki = 12 nM T32060 D01NTM 11264955 Ki = 53 nM T32060 D01PYU 9821248 Ki = 59 nM T32060 D01SJL 135509961 Ki = 12 nM T32060 D01TSX 9840090 Ki = 0.65 nM T32060 D01WNO 21868720 Ki = 58 nM T32060 D01XZI 10015055 Ki = 470 nM T32060 D02ESW 107992 EC50 = 420 nM T32060 D02GNN 119812 Ki = 1498 nM T32060 D02JPD 18354719 Ki = 28 nM T32060 D02RAY 16754 Ki = 966 nM T32060 D02SDX 151221 Ki = 1636 nM T32060 D02UWB 1809 Ki < 5011.87 nM T32060 D02YNH 9901086 EC50 = 75.86 nM T32060 D02YSX 197033 Ki = 61.66 nM T32060 D03DET 10287730 Ki < 2511.89 nM T32060 D03DLZ 6089 Ki = 65 nM T32060 D03IWX 44580317 Ki = 1367 nM T32060 D03NRJ 10871642 Ki = 15 nM T32060 D03TDN 1342 IC50 = 62 nM T32060 D03TSY 24825775 Ki > 1000 nM T32060 D03VUU 44521012 Ki = 92 nM T32060 D04AQE 1833 EC50 = 0.503 nM T32060 D04AZE 3277600 Ki < 6309.57 nM T32060 D04QRS 27559 Ki = 19 nM T32060 D04SCQ 3015863 Ki = 2589 nM T32060 D04UCV 14595512 Ki = 320 nM T32060 D04YCJ 135399866 Ki = 5.8 nM T32060 D05DAG 164682 EC50 = 2.64 nM T32060 D05EQG 5265 Ki = 1.1 nM T32060 D05JIO 9859429 Ki = 82 nM T32060 D05NWH 443390 Ki = 125.89 nM T32060 D05RKS 20293994 Ki = 754 nM T32060 D05SWY 44404899 Ki = 923 nM T32060 D05ULV 44580318 Ki = 124 nM T32060 D05XGR 6918647 Ki = 1258.93 nM T32060 D05YFZ 44373221 Ki = 480 nM T32060 D05ZUX 44207909 Ki >= 1000 nM T32060 D06ABJ 11492162 Ki = 335 nM T32060 D06PKJ 62787 Ki = 211 nM T32060 D06VDN 443391 IC50 = 32.4 nM T32060 D07CZJ 44447998 Ki = 92 nM T32060 D07ETF 9838960 Ki = 4.7 nM T32060 D07GBV 10091189 Ki = 0.48 nM T32060 D07GQP 11477180 Ki = 62.4 nM T32060 D07LRJ 5312149 Ki = 1740 nM T32060 D07XTU 1229 Ki = 0.46 nM T32060 D08CKM 9863250 Ki < 5011.87 nM T32060 D08CZT 9882067 Ki = 12 nM T32060 D08DOG 25130235 Ki = 4100 nM T32060 D08EFH 36906 Ki = 4.6 nM T32060 D08FUK 10845306 Ki = 794 nM T32060 D08GJS 44404906 Ki = 982 nM T32060 D08JCU 44439386 Ki = 7.7 nM T32060 D08MNG 16086368 Ki = 53 nM T32060 D08OFG 11177588 Ki = 1930 nM T32060 D08VGJ 9904281 Ki = 434 nM T32060 D08XGI 10379653 Ki = 9.6 nM T32060 D08ZWM 4980 EC50 = 24 nM T32060 D09BNS 439280 EC50 = 1.349 nM T32060 D09HFT 44439376 Ki = 7.4 nM T32060 D09HJL 10331436 Ki = 2 nM T32060 D09OYA 2107 EC50 = 2 nM T32060 D09PIN 3378093 Ki = 1584.89 nM T32060 D09RPR 16737207 Ki > 10000 nM T32060 D09WIL 10028436 Ki = 63.1 nM T32060 D0A6LB 46228433 EC50 = 2202 nM T32060 D0AP6N 44404886 EC50 = 32 nM T32060 D0B0PP 79698 Ki > 10000 nM T32060 D0B1GJ 44578927 Ki = 109 nM T32060 D0B1KT 15953802 Ki = 100000000 nM T32060 D0B3WX 5475158 Ki = 13 nM T32060 D0B9ZK 25138699 Ki = 7.5 nM T32060 D0C1SE 14595509 Ki = 635 nM T32060 D0C2UJ 8974 Ki > 10000 nM T32060 D0C3EX 1797 Ki = 260 nM T32060 D0C5XQ 1832 Ki = 15 nM T32060 D0C7FL 77575 Ki = 4140 nM T32060 D0CK9K 6918513 IC50 = 620 nM T32060 D0D8GV 9830741 Ki > 500 nM T32060 D0D9YW 3292447 Ki = 50.12 nM T32060 D0DY5G 443389 Ki = 398.11 nM T32060 D0E3AL 56597938 Ki = 0.6 nM T32060 D0E6NW 9859257 EC50 = 62 nM T32060 D0F0IA 11301655 Ki = 370 nM T32060 D0F1FN 15893127 Ki = 600 nM T32060 D0F5WP 135520431 Ki = 20 nM T32060 D0F6CD 5202 EC50 = 0.27 nM T32060 D0FF6S 16038374 IC50 = 3000 nM T32060 D0FL1D 9842124 Ki = 20 nM T32060 D0FU5E 10220053 Ki > 1000 nM T32060 D0G7LE 10991121 Ki = 1.2 nM T32060 D0G7QT 10131112 IC50 = 240 nM T32060 D0G8CV 9954003 Ki = 19.95 nM T32060 D0G8VU 3645619 Ki = 4010 nM T32060 D0GI7S 3146743 Ki > 10000 nM T32060 D0H2WQ 54562 Ki = 25000 nM T32060 D0H3WJ 44435193 Ki = 180 nM T32060 D0H5XR 3045225 Ki = 13 nM T32060 D0H7PC 6918553 Ki > 7943.28 nM T32060 D0H9QG 5312148 Ki < 15848.93 nM T32060 D0I2WQ 44579031 Ki = 95 nM T32060 D0I9RW 135427931 Ki = 21 nM T32060 D0J2ID 10730997 Ki = 794 nM T32060 D0J2UA 135433933 Ki = 2000 nM T32060 D0J6JT 1355 EC50 = 7.2 nM T32060 D0J8RI 9964324 Ki = 158.49 nM T32060 D0K5NZ 68848 Ki = 19.95 nM T32060 D0K6VR 44287208 Ki = 330 nM T32060 D0K8DY 44373281 Ki = 721 nM T32060 D0K8ZZ 448222 Ki > 10000 nM T32060 D0K9WJ 11324846 IC50 > 10000 nM T32060 D0KS0I 24894910 EC50 > 10000 nM T32060 D0KU6D 10679289 Ki = 251 nM T32060 D0L0MU 209436 Ki = 4130 nM T32060 D0L5MW 181743 Ki = 832 nM T32060 D0L8MR 4076 Ki = 551 nM T32060 D0M1YU 10198431 Ki = 31 nM T32060 D0M3PV 133633 Ki = 695 nM T32060 D0M5ZE 5311416 Ki = 501.19 nM T32060 D0N8YG 135414348 Ki = 1.8 nM T32060 D0ND5D 10493741 Ki = 14 nM T32060 D0NM6R 135412764 Ki = 1700 nM T32060 D0O5KK 44451373 Ki = 99 nM T32060 D0OG0R 10337743 IC50 = 351 nM T32060 D0PC7A 10106214 Ki = 100 nM T32060 D0Q1ZC 9838958 Ki = 7.8 nM T32060 D0Q3OK 9855823 Ki = 199.53 nM T32060 D0Q6PI 1001 Ki = 16800 nM T32060 D0Q9FU 10330734 Ki = 12 nM T32060 D0Q9KP 44452853 Ki = 89 nM T32060 D0R3GW 10296414 Ki = 3162.28 nM T32060 D0R5WB 9817960 Ki = 2.6 nM T32060 D0R8PL 44579030 Ki = 109 nM T32060 D0R8VT 44404883 EC50 = 633 nM T32060 D0RC9T 9795587 Ki = 0.99 nM T32060 D0S0WX 10354158 Ki = 32 nM T32060 D0S3WR 120445 Ki = 1151 nM T32060 D0T2RY 9948320 Ki >= 1000 nM T32060 D0T7RY 9813197 Ki = 93 nM T32060 D0T8UR 44404904 Ki = 498 nM T32060 D0U3GZ 98527 Ki = 0.66 nM T32060 D0U5HQ 44287445 Ki = 1040 nM T32060 D0U7BH 9815618 EC50 = 199.53 nM T32060 D0U7UD 10826147 Ki = 2511.89 nM T32060 D0U9HE 3693566 Ki = 630.96 nM T32060 D0V5SQ 68186 IC50 = 0.3162 nM T32060 D0V7OO 10386282 IC50 = 4400 nM T32060 D0W8EB 44404905 Ki = 588 nM T32060 D0XX7J 44451369 Ki = 46 nM T32060 D0Y0SA 135399666 Ki = 105 nM T32060 D0Y9TL 13702393 Ki = 1164 nM T32060 D0YZ3E 44435200 Ki = 1600 nM T32060 D0ZZ4S 44580316 Ki = 1158 nM T32060 D0ZZ4Z 21854226 Ki = 429 nM T53764 D02EYG 10096344 IC50 = 70.8 nM T53764 D0L3DK 6918537 IC50 = 3720 nM T53764 D0NJ5H 11450633 IC50 > 100000 nM T53764 D0T8XB 44513473 IC50 = 72700 nM T53764 D0U2JP 4369359 IC50 = 5830 nM T53764 D04XIO 11253490 IC50 = 7520 nM T53764 D07HZG 11516136 IC50 = 10300 nM T53764 D0FQ2U 6918572 IC50 = 66 nM T53764 D0M3XR 46209133 IC50 > 67000 nM T53764 D0K2ZQ 57378228 IC50 = 367 nM T53764 D0A1NU 16049769 Ki > 30000 nM T53764 CV87XC 9835734 Ki = 14639 nM T53764 C8XO1Z 9859008 Ki > 23440 nM T53764 C5CZ6J 9865563 Ki > 23440 nM T53764 CZ1S9O 9942554 IC50 = 11 nM T53764 C83ZDL 10096130 IC50 > 35000 nM T53764 CKY4R8 10112957 Ki > 23440 nM T53764 C0Q7BK 10127057 IC50 > 10000 nM T53764 CLZF79 10133903 Ki = 19076 nM T53764 C2RW5Z 10135822 Ki > 23440 nM T53764 CUE7K0 10156677 Ki > 23440 nM T53764 CUB1G7 10157334 Ki = 9450 nM T53764 C6PZ1U 10160012 Ki = 16980 nM T53764 C0L1KV 10162433 Ki = 20395 nM T53764 C29RUO 10162817 Ki = 9660 nM T53764 C6S5OX 10179212 Ki > 23440 nM T53764 CF7C3M 10180260 Ki = 15776 nM T53764 C05DXJ 10200731 Ki > 23440 nM T53764 C6ISW4 10203198 Ki = 12380 nM T53764 CD2U3A 10203599 Ki > 23440 nM T53764 CBZ3P2 10221723 Ki > 23440 nM T53764 CBC45I 10222923 Ki > 23440 nM T53764 CZ92XV 10225547 Ki > 23440 nM T53764 C5P0AO 10238227 IC50 > 10000 nM T53764 CQ07AR 10270647 Ki = 9660 nM T53764 CD0P5E 10271196 Ki > 23440 nM T53764 CQ36IM 10272290 Ki = 12176 nM T53764 CA7Q8J 10298482 Ki = 12845 nM T53764 CY3LK8 10300368 Ki = 6863 nM T53764 C3FB4T 10310021 IC50 > 10000 nM T53764 CQ7J2Z 10383508 IC50 > 100000 nM T53764 CWCA76 10439426 IC50 = 21000 nM T53764 C4OC6P 10455620 IC50 > 10000 nM T53764 C1WKE4 10455621 IC50 > 10000 nM T53764 CH1DG5 10478099 IC50 > 10000 nM T53764 C1WG0P 10798659 IC50 = 11 nM T53764 CF1LD8 11199808 Ki = 2200 nM T53764 CHX25W 11232123 IC50 > 100000 nM T53764 CYL67P 11232890 Ki = 479 nM T53764 CDLT06 11245133 IC50 > 10000 nM T53764 CKL1A8 11268930 Ki = 536 nM T53764 CM0YI7 11269397 Ki = 240 nM T53764 CEZ27P 11314348 Ki = 505 nM T53764 CW3QZ7 11374531 IC50 = 740 nM T53764 C30JEU 11381416 IC50 > 30000 nM T53764 CL9HN3 11395030 Ki = 888 nM T53764 CTW02K 11406276 Ki = 1770 nM T53764 CV1E7C 11406559 IC50 > 10000 nM T53764 CY15PU 11429829 Ki = 394 nM T53764 CTD0S4 11486251 Ki = 1527 nM T53764 C06RUA 11493219 IC50 > 30000 nM T53764 CAH5Z6 11500899 IC50 > 30000 nM T53764 CW38YC 11507527 IC50 > 10000 nM T53764 C7CLT9 11515196 IC50 > 10000 nM T53764 C2TCM8 11523077 IC50 = 7000 nM T53764 CMYN65 11526865 IC50 > 40000 nM T53764 CZ35WN 11533932 IC50 > 40000 nM T53764 CG7I8Z 11538992 IC50 = 60000 nM T53764 CPR71X 11540951 IC50 > 40000 nM T53764 C98GDW 11541277 IC50 > 40000 nM T53764 CBR9K8 11541314 IC50 > 40000 nM T53764 C9I5GV 11551088 IC50 > 10000 nM T53764 CCFP45 11558852 IC50 > 10000 nM T53764 CMN2K0 11566106 IC50 > 20000 nM T53764 CI5W4Y 11566450 IC50 > 30000 nM T53764 CY0A7J 11570138 IC50 > 40000 nM T53764 CAE39I 11573427 IC50 > 30000 nM T53764 CQU80H 11576569 IC50 > 40000 nM T53764 CW94NS 11577331 IC50 > 40000 nM T53764 CQ86GI 11577431 IC50 > 40000 nM T53764 CJV39M 11579395 Ki = 23 nM T53764 CAZL49 11584650 IC50 > 40000 nM T53764 C5JYV7 11591936 IC50 > 40000 nM T53764 CDE3P6 11594121 IC50 > 10000 nM T53764 C9MXO0 11596219 IC50 > 20000 nM T53764 C15DLO 11608317 IC50 > 33000 nM T53764 CQL5S8 11613750 IC50 > 40000 nM T53764 CD3YU1 11616861 IC50 > 30000 nM T53764 C2APG7 11623550 IC50 > 30000 nM T53764 CR8XO2 11623606 IC50 > 10000 nM T53764 CDZ72J 11624893 IC50 > 20000 nM T53764 C7YKC0 11628195 IC50 > 40000 nM T53764 C5P3NB 11644467 IC50 > 10000 nM T53764 C3RZO9 11645337 IC50 > 20000 nM T53764 CXG1B4 11649741 IC50 > 40000 nM T53764 C3Y7EL 11678025 IC50 > 40000 nM T53764 CNF1M4 11681778 IC50 = 7951 nM T53764 C8SI4E 11702902 IC50 > 20000 nM T53764 CIEJ54 11720809 IC50 > 40000 nM T53764 C13JIX 15949418 IC50 = 8800 nM T53764 C49NUJ 15949507 IC50 = 10600 nM T53764 C8M0FT 15951543 IC50 = 650 nM T53764 CI3DB4 15951636 Ki = 7.9 nM T53764 C8QRV9 15951839 Ki = 142 nM T53764 CMNT83 15951928 Ki = 751 nM T53764 C13-MAR 16040457 IC50 = 610 nM T53764 CS7DQ3 16090844 Ki > 30000 nM T53764 C8CVG9 16090856 Ki > 30000 nM T53764 CA1PV5 16216352 IC50 > 33000 nM T53764 CD9MQ6 16223559 IC50 > 20000 nM T53764 CQ7G8T 16223560 IC50 = 175 nM T53764 CN24YP 16223762 IC50 > 20000 nM T53764 CF37TH 16226604 IC50 = 10352 nM T53764 C6ANU2 16226605 IC50 = 16985 nM T53764 C61RFP 16755651 IC50 = 1410 nM T53764 C0X4SO 22029457 IC50 > 100000 nM T53764 CLK4G6 22029894 IC50 > 100000 nM T53764 C9Y1BP 23646016 IC50 = 13609 nM T53764 CL8DY2 23646017 IC50 > 20000 nM T53764 CT6Q1R 23646018 IC50 = 8803 nM T53764 C8VS1X 23646019 IC50 = 5129 nM T53764 CL4BX5 23646020 IC50 > 20000 nM T53764 CZ24WC 23646021 IC50 > 20000 nM T53764 C98VYW 23646022 IC50 > 20000 nM T53764 CCL17M 23646023 IC50 > 20000 nM T53764 CT16HE 23646024 IC50 = 19478 nM T53764 CVSH12 23646026 IC50 > 100000 nM T53764 CNP9T1 24180585 IC50 > 30000 nM T53764 CX8DH1 24769723 IC50 = 22000 nM T53764 C0H8OB 24776705 IC50 > 10000 nM T53764 C24GLZ 24776939 IC50 > 10000 nM T53764 C6LD2J 24777439 IC50 > 10000 nM T53764 CK8EL5 24777568 IC50 > 10000 nM T53764 CQ20PV 24777692 IC50 > 10000 nM T53764 C1WF3I 24777804 IC50 > 10000 nM T53764 C29SZR 24784416 IC50 > 100000 nM T53764 CUM03S 24798754 IC50 = 30000 nM T53764 CYL69J 24951732 IC50 = 62000 nM T53764 CNP3T1 24951733 IC50 = 16000 nM T53764 CDCP18 24952087 IC50 = 3300 nM T53764 CIM7S2 24952089 IC50 = 58000 nM T53764 C7IDX9 25132160 IC50 = 22000 nM T53764 CSU0B5 25189891 Ki > 30000 nM T53764 C60SVD 42636924 IC50 > 20000 nM T53764 CS40ML 44123747 IC50 > 50000 nM T53764 CFY7P3 44360924 IC50 > 35000 nM T53764 CRO16Q 44403360 IC50 = 4100 nM T53764 C0FC7D 44403361 IC50 = 6800 nM T53764 C3TOY4 44403392 IC50 = 24000 nM T53764 CU39LX 44403393 IC50 = 6500 nM T53764 CIA8Y3 44403397 IC50 = 290 nM T53764 C6P7NE 44403398 IC50 = 530 nM T53764 CP34SF 44403405 IC50 = 4.6 nM T53764 C60VBT 44403406 IC50 = 270 nM T53764 CQ5T4Y 44403412 IC50 = 7800 nM T53764 CMX9B1 44403416 IC50 = 99 nM T53764 CUKG07 44403417 IC50 = 770 nM T53764 CX29FU 44403421 IC50 = 37000 nM T53764 C2P4CQ 44403422 IC50 = 150 nM T53764 C4YAH3 44404393 IC50 = 180 nM T53764 C02SYC 44406179 Ki = 7925 nM T53764 CU8B3S 44406189 Ki = 1276 nM T53764 C5P1RX 44406284 Ki = 5158 nM T53764 C8LC2A 44418213 IC50 > 20000 nM T53764 CTM1Y8 44418214 IC50 > 20000 nM T53764 C1EMA5 44418215 IC50 > 20000 nM T53764 CWDH12 44418216 IC50 > 20000 nM T53764 C1FB4K 44418218 IC50 > 20000 nM T53764 CVC3R4 44418219 IC50 > 20000 nM T53764 CU1FG2 44418222 IC50 > 20000 nM T53764 C8ZH5R 44418223 IC50 > 20000 nM T53764 CA9YM3 44418225 IC50 > 20000 nM T53764 CQE5Y0 44418229 IC50 > 20000 nM T53764 CID62U 44418230 Ki = 51 nM T53764 CI2H7Q 44418231 Ki = 20 nM T53764 C2LXS7 44418232 IC50 > 20000 nM T53764 CXCV19 44418233 Ki = 14 nM T53764 CZW38C 44418239 Ki = 29 nM T53764 C7KF0X 44418240 Ki = 161 nM T53764 C8QJ7H 44418242 Ki = 265 nM T53764 C60KPZ 44418243 Ki = 191 nM T53764 CMKW39 44418246 Ki = 146 nM T53764 CEBQ24 44418249 Ki = 246 nM T53764 CVP72G 44418250 Ki = 350 nM T53764 C59HZQ 44418251 Ki = 7.5 nM T53764 CDX2Q5 44418253 Ki = 94 nM T53764 C0RV8O 44418254 Ki = 2900 nM T53764 C37KEO 44418255 Ki = 12 nM T53764 C2UR9X 44418256 IC50 > 20000 nM T53764 CK20CA 44418257 IC50 > 20000 nM T53764 CO3GL6 44418260 IC50 > 20000 nM T53764 CY3O7C 44418261 IC50 > 20000 nM T53764 C0ITV9 44418262 IC50 > 20000 nM T53764 C68SHD 44418264 IC50 > 20000 nM T53764 CDI98V 44418265 IC50 > 20000 nM T53764 CHO5P1 44418266 IC50 > 20000 nM T53764 C95XQC 44418268 IC50 > 20000 nM T53764 CR0A1M 44431316 IC50 = 60000 nM T53764 CV1R7A 44431317 IC50 > 100000 nM T53764 C08ZST 44440659 Ki > 30000 nM T53764 CR3PM7 44440662 Ki > 30000 nM T53764 CB4Q0H 44440663 Ki > 30000 nM T53764 CCSI57 44440665 Ki > 30000 nM T53764 CSN27E 44445042 IC50 > 10000 nM T53764 CGN61Q 44445047 IC50 > 10000 nM T53764 CYW8E3 44445051 IC50 > 10000 nM T53764 CRG64M 44445053 IC50 > 10000 nM T53764 C6ZID3 44445055 IC50 > 10000 nM T53764 C72KOR 44445057 IC50 > 10000 nM T53764 C0RTA6 44445060 IC50 > 10000 nM T53764 CIK8G3 44445063 IC50 > 10000 nM T53764 CN05VX 44445065 IC50 > 10000 nM T53764 COA90R 44445067 IC50 > 10000 nM T53764 C1U4YQ 44565237 IC50 > 20000 nM T53764 CRK69O 44565238 IC50 > 20000 nM T53764 C6M2WD 44565239 IC50 > 20000 nM T53764 CTZ9L0 44565254 IC50 > 20000 nM T53764 CEMV93 44565274 IC50 > 20000 nM T53764 C5E6PQ 44565275 IC50 = 13000 nM T53764 CI93OK 44565276 IC50 > 20000 nM T53764 C2HRF1 44565277 IC50 = 590 nM T53764 CFEC28 44565466 IC50 > 20000 nM T53764 C5MON6 44565467 IC50 > 20000 nM T53764 CGA4U6 44565488 IC50 > 20000 nM T53764 C1BZ3I 44565489 IC50 > 20000 nM T53764 CP3C5F 44565490 IC50 > 20000 nM T53764 CRU86T 44565491 IC50 > 20000 nM T53764 C3C2DL 44565492 IC50 > 20000 nM T53764 CJ2W1P 44565512 IC50 > 20000 nM T53764 C5Z9GW 44565513 IC50 > 20000 nM T53764 C3I0MO 44565514 IC50 > 20000 nM T53764 CI3J6Y 44565535 IC50 > 20000 nM T53764 CB90XZ 44565536 IC50 > 20000 nM T53764 C01SLH 44565537 IC50 > 20000 nM T53764 C8Y2LX 44565538 IC50 > 20000 nM T53764 CXD19F 44565539 IC50 > 20000 nM T53764 CTC24F 44590734 IC50 = 46 nM T53764 CI0FT1 44593463 IC50 > 20000 nM T53764 CK5P9W 45269994 IC50 > 10000 nM T53764 C2EK3O 45273409 IC50 > 10000 nM T53764 CDP7Q4 46870369 IC50 = 350 nM T53764 CAL9K6 46891534 IC50 > 20000 nM T53764 C4XTW7 46893990 IC50 = 79 nM T53764 C8DSG7 46916343 IC50 = 510 nM T53764 C3RO8F 46916345 IC50 = 200 nM T53764 CX07LJ 46916346 IC50 > 20000 nM T53764 CF94MW 46916347 IC50 = 3200 nM T53764 CH3F7O 46916384 IC50 = 650 nM T53764 CM8W6E 46916385 IC50 = 73 nM T53764 C6FA9Q 46916386 IC50 = 15000 nM T53764 CAW86J 46916387 IC50 > 50000 nM T53764 C63HBE 46916388 IC50 = 210 nM T53764 CD1CZ7 46916389 IC50 = 59 nM T53764 CH80LK 46916433 IC50 = 110 nM T53764 CN4A3P 46916435 IC50 = 63 nM T53764 CUQ86M 46917047 IC50 = 20 nM T53764 CS5X9L 46917048 Ki = 1.3 nM T53764 CZP24U 46917049 IC50 = 31 nM T53764 CGMJ52 46938499 IC50 > 100000 nM T53764 C5RAS7 46938602 IC50 > 100000 nM T53764 C3B1LX 46938704 IC50 = 66 nM T53764 C5TU1F 46938705 IC50 = 88 nM T53764 CAGP83 46938706 IC50 = 250 nM T53764 CP9V8Q 46938799 IC50 = 730 nM T53764 CAB2H9 46938802 IC50 > 100000 nM T53764 C80RAT 47370344 IC50 > 100000 nM T53764 CZ7A9E 49796933 IC50 > 100000 nM T53764 C5RF0Y 49796938 IC50 > 100000 nM T53764 CE0C3Y 49796939 IC50 > 100000 nM T53764 CI4ZE6 49796940 IC50 > 100000 nM T53764 CBD8K2 49796942 IC50 > 100000 nM T53764 CI25XP 49796945 IC50 > 100000 nM T53764 C8WYA5 49796953 IC50 = 21000 nM T53764 CQH86V 49796955 IC50 = 48000 nM T53764 C85CEJ 51346970 IC50 > 35000 nM T53764 C4PFT3 51346971 IC50 > 35000 nM T53764 C7RJM9 52945660 IC50 = 54 nM T53764 CC56BV 52946866 IC50 > 20000 nM T53764 CYC69Q 53317564 IC50 > 35000 nM T53764 C0QOV9 53317565 IC50 > 35000 nM T53764 CURC70 53317566 IC50 > 35000 nM T53764 C3ZK1W 53317575 IC50 > 35000 nM T53764 CBQ0J7 53317579 IC50 > 35000 nM T53764 CIY9F7 53317580 IC50 > 35000 nM T53764 C5DMS9 53317581 IC50 > 35000 nM T53764 C1XD9W 53317582 IC50 > 35000 nM T53764 CR0O8T 53317583 IC50 > 35000 nM T53764 C9GLH7 53318841 IC50 > 35000 nM T53764 C06TDE 53318842 IC50 > 35000 nM T53764 C73TER 53318856 IC50 > 35000 nM T53764 CC56NE 53318863 IC50 > 35000 nM T53764 C4UJI8 53318864 IC50 > 35000 nM T53764 C8CZ2A 53318865 IC50 > 35000 nM T53764 CLVY47 53318866 IC50 > 35000 nM T53764 CM7S5W 53319067 IC50 > 35000 nM T53764 C1X3NE 53320178 IC50 > 35000 nM T53764 C1P8BK 53320179 IC50 > 35000 nM T53764 C50UBZ 53320180 IC50 > 35000 nM T53764 C2JTR7 53320181 IC50 > 35000 nM T53764 C0TYJ5 53320182 IC50 > 35000 nM T53764 C7RSX2 53320183 IC50 > 35000 nM T53764 C9XGE4 53321472 IC50 > 35000 nM T53764 CY0ZV9 53321485 IC50 > 35000 nM T53764 CK0OB2 53321486 IC50 > 35000 nM T53764 CNK34J 53321487 IC50 > 35000 nM T53764 C7EO3D 53321495 IC50 > 35000 nM T53764 C3M7PQ 53321496 IC50 > 35000 nM T53764 C0NUQ7 53321497 IC50 > 35000 nM T53764 C31DSJ 53321498 IC50 > 35000 nM T53764 C2ZKV9 53321499 IC50 > 35000 nM T53764 C3QT0R 53321621 IC50 > 35000 nM T53764 CXIS21 53322758 IC50 > 35000 nM T53764 CY71QL 53322814 IC50 > 35000 nM T53764 CLU96Y 53322820 IC50 > 35000 nM T53764 C8YVF1 53322821 IC50 > 35000 nM T53764 C4QS6V 53322822 IC50 > 35000 nM T53764 C62JTB 53322823 IC50 > 35000 nM T53764 CT14FU 53322824 IC50 > 35000 nM T53764 CXJ1F8 53322825 IC50 > 35000 nM T53764 C3K1VY 53322826 IC50 > 35000 nM T53764 C9N6HK 53322952 IC50 > 35000 nM T53764 C9LU8M 53324129 IC50 > 35000 nM T53764 CCY7M0 53324130 IC50 > 35000 nM T53764 C4F1QK 53324142 IC50 > 35000 nM T53764 CZN71C 53324143 IC50 > 35000 nM T53764 CG83JZ 53324144 IC50 > 35000 nM T53764 CE8J1D 53324145 IC50 > 35000 nM T53764 C0Y3AC 53324153 IC50 > 35000 nM T53764 C9O1IW 53324154 IC50 > 35000 nM T53764 CTW5G0 53324155 IC50 > 35000 nM T53764 C2DPZ0 53324156 IC50 > 35000 nM T53764 CSN28M 53324293 IC50 > 35000 nM T53764 C25OJW 53325399 IC50 > 35000 nM T53764 CXW5O9 53325446 IC50 > 35000 nM T53764 C1SO0C 53325447 IC50 > 35000 nM T53764 C1S3WB 53325453 IC50 > 35000 nM T53764 C2KFW6 53325454 IC50 > 35000 nM T53764 C4ZFR5 53325455 IC50 > 35000 nM T53764 CV0H8P 53326691 IC50 > 35000 nM T53764 C3ZWN6 53326704 IC50 > 35000 nM T53764 C73SKG 53326705 IC50 > 35000 nM T53764 CG9V4W 53326706 IC50 > 35000 nM T53764 C5K8CP 53326713 IC50 > 35000 nM T53764 C0P8KM 57397016 IC50 = 1000 nM T53764 CX31VN 57403989 IC50 = 4700 nM T53764 CXRS60 57406622 IC50 = 88335 nM T53764 CNOX18 57406623 IC50 = 9920 nM T53764 CZS03L 57406803 IC50 = 268 nM T53764 C80RBH 57406804 IC50 > 50000 nM T53764 CMH17V 57406805 IC50 = 755 nM T53764 C2EX0S 57406806 IC50 = 4620 nM T53764 CR6QP4 57406990 IC50 = 4640 nM T53764 CFML71 57406991 IC50 = 3122 nM T53764 C2PX9N 57406992 IC50 = 22406 nM T53764 C0COE1 57407188 IC50 = 78508 nM T53764 C5G3KT 57407189 IC50 > 100000 nM T53764 C8MJK5 57407191 IC50 = 14740 nM T53764 CVS34M 57407192 IC50 = 3052 nM T53764 C7AZB3 57407370 IC50 = 15288 nM T53764 C9ZE7J 58874273 IC50 = 30600 nM T53764 C4AY5G 60195086 IC50 > 100000 nM T53764 CIY07P 60195087 IC50 > 100000 nM T53764 CB9E2P 60195088 IC50 > 100000 nM T53764 CH3Z7F 68658979 IC50 = 4100 nM T53764 C6HRX1 68845950 IC50 > 100000 nM T53764 C5W6LY 70681316 IC50 > 10000 nM T53764 CVYH31 70689717 IC50 > 10000 nM T53764 CP6G5W 71203746 IC50 > 100000 nM T53764 C32UMV 71203748 IC50 = 16300 nM T53764 C04XQY 71203752 IC50 > 100000 nM T53764 CIQ7O2 71203767 IC50 = 7300 nM T53764 C7LKV0 71203783 IC50 = 53600 nM T53764 C7B8AO 71621488 IC50 = 3.3 nM T53764 C8T2PW 71655265 IC50 = 0.47 nM T53764 C1HGS0 71655267 IC50 = 54 nM T53764 C9XJ6S 71655268 IC50 = 500 nM T53764 CX6AI5 71655326 IC50 = 3.4 nM T53764 C9H0QK 71655327 IC50 = 16 nM T53764 CLM0G6 71655328 IC50 = 9.4 nM T53764 CFS59P 71655329 IC50 = 6.4 nM T53764 CZL7N9 71655330 IC50 = 120 nM T53764 CR7I0Y 71655331 IC50 = 350 nM T53764 CLCH69 71655332 IC50 = 65 nM T53764 CL0ZS6 71655390 IC50 = 15 nM T53764 C6Y9LQ 71655391 IC50 = 1300 nM T53764 C93CXQ 71655392 IC50 = 1100 nM T53764 C8P1GB 71655393 IC50 = 9300 nM T53764 CVB75Q 71655394 IC50 = 1.1 nM T53764 CH4ZS0 71655395 IC50 > 100000 nM T53764 C1HL2A 72188903 IC50 = 51000 nM T53764 CLS1A0 72188904 IC50 > 100000 nM T53764 CL7P3D 72193502 IC50 > 100000 nM T53764 C4AXB8 72193503 IC50 > 100000 nM T53764 CQC28P 72193504 IC50 > 6400 nM T53764 CV87PE 72193505 IC50 > 100000 nM T53764 C65DFP 72697059 IC50 = 2220 nM T53764 CZ56DO 72697061 IC50 = 1580 nM T53764 C1A2KX 72697062 IC50 = 1460 nM T53764 CS5U1F 72697063 IC50 = 2140 nM T53764 CWNZ91 72697207 IC50 = 800 nM T53764 C6BWI4 72697208 IC50 = 7870 nM T53764 C9JA1Q 72697209 IC50 = 3010 nM T53764 CF6A8N 72697210 IC50 = 2690 nM T53764 CTMR03 72697211 IC50 = 5810 nM T53764 CP9NV5 72697212 IC50 = 27630 nM T53764 C1P8HS 72697352 IC50 = 2600 nM T53764 CC7G3M 72697353 IC50 = 1580 nM T53764 CAXV78 72697355 IC50 = 1530 nM T53764 CGV09W 72697356 IC50 = 82 nM T53764 CIF9D7 72697357 IC50 = 470 nM T53764 CC8RA6 72697358 IC50 = 140 nM T53764 C1EC7S 72697359 IC50 = 3650 nM T53764 C8CRO6 72697494 IC50 = 470 nM T53764 C03NKY 72697495 IC50 = 610 nM T53764 CP0MU3 72697496 IC50 = 1700 nM T53764 CI60AK 72697497 IC50 = 140 nM T53764 CO19YK 72697498 IC50 = 3910 nM T53764 C47IGZ 72697499 IC50 = 6100 nM T53764 C65OPG 72697500 IC50 = 150 nM T53764 C3ZP7N 72697501 IC50 = 220 nM T53764 C7EF8C 72697646 IC50 = 900 nM T53764 CSZR98 73346173 IC50 > 100000 nM T53764 C1L4RX 73346174 IC50 > 6400 nM T53764 CGNL10 73347698 IC50 > 100000 nM T53764 CO5TB8 73349220 IC50 > 100000 nM T53764 CNC6B8 73350798 IC50 > 100000 nM T53764 CDBV29 73350799 IC50 > 100000 nM T53764 CYG04J 73352283 IC50 > 100000 nM T53764 CV6BA3 73353756 IC50 > 100000 nM T53764 C51QGP 73353757 IC50 = 75000 nM T53764 CBK37N 73353758 IC50 > 100000 nM T53764 CLO76J 73355285 IC50 > 100000 nM T53764 CCVT96 73355286 IC50 > 100000 nM T53764 CIV7Y8 89668929 IC50 > 10000 nM T53764 CBQ38C 101879512 IC50 = 34180 nM T53764 CM7E4V 101887269 IC50 = 1900 nM T53764 C8EH0J 101887270 IC50 = 1800 nM T53764 CDT67J 101887271 IC50 = 1200 nM T53764 C4F2CS 101887272 IC50 = 5800 nM T53764 C58XWA 101887273 IC50 = 3300 nM T53764 C3Y9ET 101887274 IC50 > 10000 nM T53764 C1AF8C 101887275 IC50 > 50000 nM T53764 CH7QC5 101887276 IC50 > 10000 nM T53764 CO4FR2 101887277 IC50 = 10300 nM T53764 C9JEH0 101887278 IC50 = 11000 nM T53764 C52GIO 101887279 IC50 > 12500 nM T53764 CT2MZ8 118712764 IC50 = 5900 nM T53764 C3W5RU 118712765 IC50 = 3120 nM T53764 CKA1N5 118712766 IC50 = 1090 nM T53764 C8M6ZW 118712767 IC50 = 6850 nM T53764 CV5C6D 118712768 IC50 = 5770 nM T53764 C2NSC7 118712769 IC50 = 2730 nM T53764 CAR4W5 118712772 IC50 = 1690 nM T53764 CRWT85 118712773 IC50 = 4830 nM T53764 C4T2FY 118712775 IC50 = 3380 nM T53764 CJ8EL0 118712778 IC50 = 34410 nM T53764 C07UOL 118712779 IC50 = 109880 nM T53764 CD0HQ4 118712781 IC50 = 153700 nM T53764 C46TMQ 118712785 IC50 = 3850 nM T53764 C5M3BX 118712788 IC50 = 12460 nM T53764 CK7HN4 118722408 IC50 = 3350 nM T53764 CK71WT 118722410 IC50 = 3290 nM T53764 CI74ZM 118722411 IC50 = 3920 nM T53764 CH1P7Y 118722412 IC50 = 1710 nM T53764 CL8TY5 118722413 IC50 = 6360 nM T53764 C8KUP0 118722416 IC50 = 2060 nM T53764 COG4V6 118722421 IC50 = 4030 nM T53764 CN78TQ 122189864 IC50 > 100000 nM T53764 CNM82F 122189865 IC50 > 100000 nM T53764 C19GHJ 122189866 IC50 > 10000 nM T53764 C3U9KC 122189867 IC50 > 100000 nM T53764 CW5V3U 122189868 IC50 = 41000 nM T53764 CCG05R 122189869 IC50 > 100000 nM T53764 CI01PT 122189870 IC50 > 100000 nM T53764 C80EWF 122189871 IC50 > 100000 nM T53764 C3N7JC 122189872 IC50 > 100000 nM T53764 CG8O1J 122189873 IC50 > 100000 nM T53764 CK0US2 122189874 IC50 > 100000 nM T53764 C5V6NI 122189875 IC50 > 100000 nM T53764 CV7A9Y 122189876 IC50 > 100000 nM T53764 CN86VR 122189878 IC50 > 50000 nM T53764 C6NIM5 127048874 IC50 = 10000 nM T53764 CXD69M 127048875 IC50 = 100000 nM T53764 C65MAC 127048876 IC50 = 91000 nM T53764 C23BWQ 127049179 IC50 = 7000 nM T53764 CNCB06 127049180 IC50 = 10000 nM T53764 CJ8SG3 127049204 IC50 = 100000 nM T53764 CRM04V 127049507 IC50 = 55000 nM T53764 C76VPA 127049823 IC50 = 2700 nM T53764 CH0X6Q 127050132 IC50 = 18000 nM T53764 CIGA32 127050759 IC50 = 4600 nM T53764 CNY90B 127050760 IC50 = 23000 nM T53764 C80WCY 127050761 IC50 = 9700 nM T53764 CUVQ34 127050762 IC50 = 77000 nM T53764 CJMS57 127051032 IC50 = 6400 nM T53764 C9V4EG 127051045 IC50 = 7600 nM T53764 C7W8JR 127051639 IC50 = 57000 nM T53764 C36SXH 127052286 IC50 = 30000 nM T53764 CBR1F8 127052287 IC50 = 24000 nM T53764 CHZX75 127052288 IC50 = 18000 nM T53764 CB34GQ 127052289 IC50 = 35000 nM T53764 CLG0Q3 127052290 IC50 = 53000 nM T53764 CL2S0F 127052581 IC50 = 570 nM T53764 C1W5AL 127052582 IC50 = 1800 nM T53764 C4TI8H 127052590 IC50 = 11000 nM T53764 CNV0A8 127052636 IC50 = 280 nM T53764 CS2Z9R 127052637 IC50 = 450 nM T53764 C75EAL 127052638 IC50 = 280 nM T53764 CR4VI2 137225025 IC50 = 1700 nM T53764 C7YP3B 155530585 IC50 = 107 nM T53764 C8EQ4C 155530631 IC50 > 100000 nM T53764 CRL47X 155559391 IC50 = 11446 nM T53764 D03DNV 71655266 Ki = 9 nM T53764 D04CAR 10607286 IC50 = 52 nM T15053 D06ACW 6083 IC50 > 500000 nM T15053 D0Z0HH 3503 Ki = 1900 nM T15053 CZ1JT5 5242 Ki > 100000 nM T15053 C3RJ7D 6844 IC50 > 500000 nM T15053 CC3YF8 120118 IC50 > 2000000 nM T15053 CEYH47 122660 Ki = 2000 nM T15053 C8W1NR 169266 IC50 = 132000 nM T15053 C92FXK 247635 IC50 > 500000 nM T15053 C2Q6NV 331941 IC50 > 500000 nM T15053 C2QIP5 444215 Ki = 188000 nM T15053 C0DHW5 467478 Ki = 2000 nM T15053 CDXR51 560735 IC50 > 500000 nM T15053 CQ59EK 596481 IC50 > 500000 nM T15053 CY52ZP 739192 IC50 > 500000 nM T15053 CFD5U6 747917 IC50 > 500000 nM T15053 CMH25I 980714 IC50 = 250 nM T15053 C5GPR0 981025 IC50 = 2300 nM T15053 CLG45C 1498318 IC50 = 22200 nM T15053 C3VSM7 1498344 IC50 = 26700 nM T15053 CC5MI8 1563320 IC50 > 500000 nM T15053 C7EX6Z 1727849 IC50 = 1240 nM T15053 CO9J4Y 1727855 IC50 > 100000 nM T15053 C7FC2X 1728053 IC50 = 3400 nM T15053 C5WJ7I 2729667 IC50 > 100000 nM T15053 C6S3OQ 3127725 IC50 = 6590 nM T15053 CSA9G1 4092653 IC50 = 22470 nM T15053 C6M9DJ 4127761 IC50 = 3500 nM T15053 CW7S2J 4141306 IC50 > 500000 nM T15053 CZ3L6A 4293432 IC50 > 500000 nM T15053 CC5HU4 5762408 Ki = 39000 nM T15053 C5UD6G 6882908 IC50 = 43000 nM T15053 C7M9PC 6917187 IC50 = 27700 nM T15053 CIM17U 7292959 EC50 = 680 nM T15053 CWJ6K9 7293051 EC50 = 3700 nM T15053 C71GCP 7293057 EC50 = 9700 nM T15053 C2PT1O 7293067 EC50 = 90 nM T15053 COI87L 7454229 IC50 > 500000 nM T15053 CZ56EW 9556853 IC50 = 37000 nM T15053 C6ZC3O 9974249 IC50 > 500000 nM T15053 C2QYA3 10093463 Ki = 200 nM T15053 CH7Y4X 10265351 Ki = 100 nM T15053 CJ3KB5 10440817 IC50 = 190700 nM T15053 CG13KM 10498042 Ki = 50 nM T15053 CRN18G 10515479 Ki = 1000 nM T15053 CYQK89 10545799 Ki = 200 nM T15053 CPU50O 10585647 Ki = 22000 nM T15053 CXF2D4 10586495 Ki = 4000 nM T15053 C0VRN5 10636040 Ki = 1000 nM T15053 C6Q5JD 10829665 Ki = 500 nM T15053 CHNQ56 11968389 IC50 = 90400 nM T15053 C72RLT 14392072 IC50 > 500000 nM T15053 C18ADR 15708693 Ki = 9100 nM T15053 C26VDI 16799813 EC50 = 12400 nM T15053 CMH16A 16803007 EC50 = 5600 nM T15053 C3N8UJ 16803010 EC50 = 270 nM T15053 C1B3UQ 16859142 EC50 = 7800 nM T15053 CX42ZS 23295347 Ki = 1000 nM T15053 CLY4V1 23605664 IC50 = 770000 nM T15053 CBXC05 24424330 IC50 = 577000 nM T15053 CIN74S 41245429 EC50 = 2140 nM T15053 C7B8CE 44259159 IC50 > 500000 nM T15053 CZO1R6 45077712 IC50 > 500000 nM T15053 CFD9U1 46893144 Ki = 4700 nM T15053 CK6LZ3 47116597 IC50 > 500000 nM T15053 CJX7U5 50940594 IC50 = 14800 nM T15053 CM3R6O 50940595 IC50 = 35900 nM T15053 C2B4IE 51354288 Ki = 10400 nM T15053 CIUC04 51354289 Ki = 19800 nM T15053 CV71WS 51355147 Ki = 5100 nM T15053 CFV0N6 51624517 EC50 = 670 nM T15053 CER7C6 52920317 Ki = 28000 nM T15053 CK5Z1U 52920321 Ki = 57000 nM T15053 C01HSL 56844251 IC50 > 500000 nM T15053 CT84SA 56844252 IC50 > 500000 nM T15053 CK3CZ5 56844253 IC50 = 1900 nM T15053 CFK30C 56844254 IC50 = 500 nM T15053 CL47WO 56844255 IC50 = 4200 nM T15053 C5W9VN 56962355 IC50 = 63.1 nM T15053 CEO0M4 57334939 IC50 = 7400 nM T15053 C0GM9Q 57340472 IC50 > 500000 nM T15053 CSZV54 57340473 IC50 = 3100 nM T15053 CZL79T 57340474 IC50 = 86200 nM T15053 CF5S0W 57340475 IC50 = 29500 nM T15053 CJ3VU7 57340476 IC50 = 290 nM T15053 C0JG4I 57340477 IC50 = 7400 nM T15053 C8S4GM 57340478 IC50 = 270 nM T15053 CADR46 70680601 IC50 = 220 nM T15053 CVQ36F 70680603 IC50 = 2200000 nM T15053 C5K4SM 71533725 IC50 = 2.6 nM T15053 C4D2VP 71562086 IC50 = 1300000 nM T15053 CLX17D 71562088 IC50 = 59000 nM T15053 C5KXA9 71562206 IC50 = 120 nM T15053 CG12TY 71562207 IC50 = 2400 nM T15053 CW3U0G 71562208 IC50 = 15200 nM T15053 C9VU5I 71562318 IC50 = 2400 nM T15053 C4YA7E 71562319 IC50 = 13000 nM T15053 CDH6E5 71562320 IC50 > 10000000 nM T15053 CN0LF5 71610855 IC50 = 16 nM T15053 C8CTI0 71615963 Ki = 37800 nM T15053 C79BIQ 71616082 Ki = 19500 nM T15053 CZP1L3 71677802 IC50 = 2000 nM T15053 CE9BS3 71719216 IC50 = 342000 nM T15053 CV4CI5 72189812 IC50 = 4000 nM T15053 CO3Z6P 72189813 IC50 > 100000 nM T15053 CI5YF7 72189814 IC50 > 100000 nM T15053 C3UK4O 72189815 IC50 > 100000 nM T15053 CH6VI2 72189816 IC50 = 24000 nM T15053 CTP06J 72189817 IC50 > 100000 nM T15053 CCE1V8 72189818 IC50 = 14000 nM T15053 CNL60P 72190137 IC50 = 10000 nM T15053 C16SNX 72190138 IC50 = 15000 nM T15053 CNIX35 72190139 IC50 = 50000 nM T15053 CL8I1Z 72190140 IC50 = 35000 nM T15053 C7RMN8 72190141 IC50 = 15000 nM T15053 CUM6L4 72190142 IC50 = 4000 nM T15053 CT2I3E 72190143 IC50 = 2000 nM T15053 CYJ56P 72190454 IC50 = 2000 nM T15053 C7B9CO 72190455 IC50 = 2000 nM T15053 CZH2C0 72190456 IC50 = 12000 nM T15053 CG98TC 72190457 IC50 > 100000 nM T15053 C2KBZ1 72190458 IC50 = 2000 nM T15053 C8F2UG 72190459 IC50 > 100000 nM T15053 CO1Z8C 72190753 IC50 > 100000 nM T15053 CDJ4B6 72190754 IC50 = 3000 nM T15053 CQ49BO 72190755 IC50 = 19000 nM T15053 C8EIZ2 72190756 IC50 > 100000 nM T15053 C9DYR3 72190758 IC50 > 100000 nM T15053 CZW4C3 72190759 IC50 = 25000 nM T15053 COM2H6 72191057 IC50 > 100000 nM T15053 C8HID5 72191058 IC50 = 73000 nM T15053 CA7Z0P 72191059 IC50 > 100000 nM T15053 C4L8BX 72191060 IC50 = 71000 nM T15053 C8KV7J 72191062 IC50 = 500 nM T15053 C4R0BA 72547453 IC50 = 15400 nM T15053 CG5SM9 72716893 EC50 = 1800 nM T15053 CI16FY 73135513 IC50 = 880 nM T15053 C79BKL 73346278 IC50 = 18000 nM T15053 CMX1W3 73348865 IC50 = 12500 nM T15053 C9H5TK 73353843 IC50 = 91000 nM T15053 CJM2V8 76148409 EC50 = 5700 nM T15053 CYRG68 78425440 IC50 > 100000 nM T15053 C8I3LH 90641413 EC50 = 3300 nM T15053 CB07HM 90667522 Ki = 45000 nM T15053 CLQ5E8 90667523 Ki = 20000 nM T15053 C2UM9N 91626457 EC50 = 4100 nM T15053 C9K7JY 91627118 EC50 = 2900 nM T15053 C2GJ0D 91629476 EC50 = 890 nM T15053 C03AGB 91664338 IC50 = 6 nM T15053 C2H7XV 91668260 IC50 = 870 nM T15053 CTD6K2 91811547 EC50 = 3400 nM T15053 CVX1H5 91814915 EC50 = 6400 nM T15053 C2CZY8 91933841 IC50 = 30 nM T15053 CWK32Y 92074669 EC50 = 340 nM T15053 CW6Y8P 92130730 EC50 = 4580 nM T15053 CBV13N 97278348 EC50 = 390 nM T15053 CND92H 99988779 IC50 = 330 nM T15053 CGVM84 118384502 IC50 = 9 nM T15053 CU59RW 118384617 IC50 = 82 nM T15053 CAN87K 118384725 IC50 = 5 nM T15053 C8VD9E 118384734 IC50 = 69 nM T15053 C9MZ5Y 118393671 IC50 = 9 nM T15053 CD35CL 118394264 IC50 = 65 nM T15053 C2LE1J 118708872 IC50 = 53000 nM T15053 CR8VJ2 118708873 IC50 = 4000 nM T15053 C60LHX 118708874 IC50 = 53000 nM T15053 CVF7S0 118708875 IC50 > 100000 nM T15053 C8RZG6 118708876 IC50 > 66000 nM T15053 C5YQ2M 118708877 IC50 > 100000 nM T15053 CH5B1T 118708878 IC50 = 36000 nM T15053 CDQ3S0 118708879 IC50 > 100000 nM T15053 CK31NM 118708880 IC50 > 100000 nM T15053 CL2VY5 118708881 IC50 = 1600 nM T15053 CT2A5M 118708882 IC50 > 100000 nM T15053 CR6OK4 118708883 IC50 > 100000 nM T15053 C2VYC3 118708884 IC50 > 100000 nM T15053 CVCS46 118708885 IC50 > 100000 nM T15053 CX8DV3 118708886 IC50 > 100000 nM T15053 CSI32O 118708887 IC50 > 100000 nM T15053 C5ELH2 118708888 IC50 > 100000 nM T15053 C6YKJ9 118708889 IC50 > 100000 nM T15053 C6Z8CK 118708890 IC50 > 100000 nM T15053 CAIM50 118708891 IC50 > 100000 nM T15053 C0YSA6 118708892 IC50 > 100000 nM T15053 CZIE63 118708893 IC50 > 100000 nM T15053 CVS79M 118708894 IC50 > 100000 nM T15053 CB38LC 118708895 IC50 > 100000 nM T15053 CVZA90 118708896 IC50 > 100000 nM T15053 C1FP6W 118708897 IC50 > 100000 nM T15053 CR9I1N 118708898 IC50 > 100000 nM T15053 CND05F 118708899 IC50 > 100000 nM T15053 CKOA17 118708900 IC50 > 100000 nM T15053 CG67IU 118708901 IC50 > 100000 nM T15053 CRXC01 118708902 IC50 > 100000 nM T15053 CM2QH9 118708903 IC50 > 100000 nM T15053 CV47ME 118708904 IC50 > 100000 nM T15053 CS8OI0 118708905 IC50 > 100000 nM T15053 CVG94O 118708906 IC50 > 100000 nM T15053 C5RG1V 118708907 IC50 > 100000 nM T15053 C5XR8F 118708908 IC50 > 100000 nM T15053 CBR62J 118708909 IC50 > 100000 nM T15053 C0NI2Q 118708910 IC50 > 100000 nM T15053 CP0GC7 118708911 IC50 > 100000 nM T15053 CR4PH2 118708912 IC50 > 100000 nM T15053 C9B8QT 118708913 IC50 > 100000 nM T15053 C71ZEN 118708914 IC50 = 63000 nM T15053 CLW6O1 118708915 IC50 = 12000 nM T15053 CLZ4D3 118708916 IC50 > 100000 nM T15053 CV9AL4 118708917 IC50 > 100000 nM T15053 CQG89R 118708918 IC50 = 24000 nM T15053 C2LIG3 118708919 IC50 > 100000 nM T15053 C26OXT 118708920 IC50 > 64000 nM T15053 CC6G9E 118708921 IC50 > 100000 nM T15053 C2G6KO 118708922 IC50 > 100000 nM T15053 C7EUJ2 118708923 IC50 > 100000 nM T15053 C8GW2O 118708924 IC50 > 100000 nM T15053 C97MQB 118708925 IC50 > 100000 nM T15053 CV8NQ5 118708926 IC50 > 100000 nM T15053 C4X5VF 118708927 IC50 > 100000 nM T15053 C6YSC4 118708928 IC50 > 100000 nM T15053 CB5F2O 118708929 IC50 > 100000 nM T15053 C1ZS0N 118708930 IC50 > 100000 nM T15053 CKU5X2 118708931 IC50 > 100000 nM T15053 C84ENI 118708932 IC50 > 100000 nM T15053 CH9Z0I 118708933 IC50 > 100000 nM T15053 C8M3JX 118708934 IC50 > 100000 nM T15053 CF29UV 118708935 IC50 > 100000 nM T15053 C40YPR 118708936 IC50 > 100000 nM T15053 CY5ST6 118708937 IC50 > 100000 nM T15053 C9W3LI 118708938 IC50 > 100000 nM T15053 CEAK31 118708939 IC50 > 100000 nM T15053 CHBD82 118708940 IC50 > 100000 nM T15053 C8GOM3 118708941 IC50 > 100000 nM T15053 C54PQF 118708942 IC50 > 100000 nM T15053 CZ6NG2 118708949 IC50 > 100000 nM T15053 C7JD3S 118708950 IC50 > 100000 nM T15053 CU78WY 118708951 IC50 > 100000 nM T15053 C5CNA6 118708952 IC50 > 100000 nM T15053 CUR2K3 118708953 IC50 > 100000 nM T15053 CT6F1W 118708954 IC50 > 100000 nM T15053 CF76ME 118708955 IC50 > 100000 nM T15053 CI34YG 118708956 IC50 > 100000 nM T15053 C1W0RM 118708957 IC50 > 100000 nM T15053 C3RL4T 118708958 IC50 > 100000 nM T15053 CYZ65E 118708959 IC50 > 100000 nM T15053 CMTN97 118708960 IC50 > 100000 nM T15053 C1BL8R 118708961 IC50 > 100000 nM T15053 CX3ZV9 118708962 IC50 > 100000 nM T15053 CBY2E6 118708963 IC50 > 100000 nM T15053 CF5IS7 118708964 IC50 > 100000 nM T15053 CY05QZ 118708965 IC50 > 100000 nM T15053 CW87RT 118708966 IC50 > 100000 nM T15053 CVM10U 118708967 IC50 = 5600 nM T15053 CUWQ40 118708968 IC50 = 5600 nM T15053 CAN71V 118708969 IC50 = 18000 nM T15053 CB9VW5 118708970 IC50 = 19000 nM T15053 COBI60 118708971 IC50 = 870 nM T15053 CP7N0R 118708972 IC50 = 3700 nM T15053 C1DA4P 118708973 IC50 = 580 nM T15053 CZT3C7 118708974 IC50 = 1000 nM T15053 CE6H7Y 118708975 IC50 = 7400 nM T15053 CIK4U6 118708976 IC50 = 270 nM T15053 CR0U5I 118708977 IC50 = 2300 nM T15053 CUT4O7 118708978 IC50 = 500 nM T15053 C93BYJ 118708979 IC50 = 15000 nM T15053 CEYN68 118708980 IC50 = 3100 nM T15053 CZ5B4K 118708981 IC50 = 6800 nM T15053 C3EDX7 118708983 IC50 = 830 nM T15053 CX7K3N 118708984 IC50 = 450 nM T15053 C3IYG8 118708985 IC50 = 640 nM T15053 CHL9D7 118708986 IC50 = 2100 nM T15053 CF7TP0 118708987 IC50 = 180 nM T15053 CU0K6S 118723134 IC50 = 4000 nM T15053 C69VGZ 118723135 IC50 = 4000 nM T15053 C1MZ5Q 118723136 IC50 = 11000 nM T15053 C4BFN5 118723137 IC50 = 26000 nM T15053 CVO7U1 118723138 IC50 = 11000 nM T15053 CY1WU8 118723139 IC50 = 13000 nM T15053 C1D0PS 118723140 IC50 = 25000 nM T15053 C0BF7E 118723141 IC50 = 66000 nM T15053 CAC13S 118723142 IC50 = 5500 nM T15053 C31VEO 118723143 IC50 = 3900 nM T15053 CCD08U 118723144 IC50 = 16000 nM T15053 CIN51G 118723145 IC50 = 5000 nM T15053 CKAJ68 118723146 IC50 = 17000 nM T15053 CDAF13 118723147 IC50 > 100000 nM T15053 C49YRS 118723148 IC50 = 9500 nM T15053 C5M1PJ 118723149 IC50 = 3800 nM T15053 C5FQ8T 118723150 IC50 = 2200 nM T15053 CL76TQ 118723151 IC50 > 100000 nM T15053 C50QSG 118723152 IC50 > 100000 nM T15053 CTUF25 118723153 IC50 = 35000 nM T15053 C7CJ3U 118723154 IC50 = 73000 nM T15053 CN9O6E 118723155 IC50 = 3500 nM T15053 CO2TC3 118723156 IC50 = 15000 nM T15053 C8G6ZQ 118723157 IC50 = 43000 nM T15053 C8XKE9 118723526 IC50 = 4100 nM T15053 CT57AW 118723527 IC50 = 13000 nM T15053 C9EF3U 118723528 IC50 = 5600 nM T15053 CC8EW9 118723529 IC50 = 46000 nM T15053 C0DO2E 118723530 IC50 = 6600 nM T15053 C0LM3H 118723531 IC50 = 7400 nM T15053 C8SHN9 118723532 IC50 = 22000 nM T15053 C1YGS7 118723533 IC50 = 59000 nM T15053 C2GHZ7 118723534 IC50 = 3300 nM T15053 CB9HQ2 118723535 IC50 = 2100 nM T15053 C1GUZ9 118723536 IC50 = 2600 nM T15053 CC34BT 118723537 IC50 = 2100 nM T15053 CT58YU 121225870 IC50 < 10 nM T15053 CTBW34 121225871 IC50 = 120 nM T15053 CXTH35 121457599 IC50 = 124 nM T15053 C2OV0L 121457603 EC50 = 3530 nM T15053 CY1JQ3 121457610 IC50 = 150 nM T15053 CIVN07 121457639 IC50 > 57000 nM T15053 CB80PQ 121457701 IC50 = 176 nM T15053 C8BIW3 121457720 IC50 > 57000 nM T15053 C8AYR7 121457742 IC50 = 17300 nM T15053 CLKW12 121457751 EC50 = 2560 nM T15053 C6ZTQ1 121457762 IC50 = 91 nM T15053 CRW7H5 121457764 IC50 > 57000 nM T15053 CSX19D 121457779 IC50 = 27700 nM T15053 CT82GB 121461607 IC50 = 53 nM T15053 C85OFV 121461678 IC50 > 57000 nM T15053 C1LDQ5 121461684 IC50 = 6230 nM T15053 CC8U4V 121461687 IC50 = 139 nM T15053 CW62PD 121461708 IC50 = 754 nM T15053 CEY1H9 121461710 IC50 = 27 nM T15053 C42KHQ 121461721 IC50 = 65 nM T15053 C2WU8I 121461723 IC50 = 95 nM T15053 CVYU65 121461728 IC50 = 42 nM T15053 C1OZ2D 121461729 IC50 = 349 nM T15053 COED87 121461743 IC50 = 19 nM T15053 C3OIR8 121461752 IC50 = 115 nM T15053 CD3KJ0 121461754 IC50 = 65 nM T15053 CT7PM0 121461757 IC50 = 57 nM T15053 CE53RH 121461760 IC50 = 144 nM T15053 C8AK4N 121461765 IC50 = 33800 nM T15053 CK9N1E 121461771 IC50 > 57000 nM T15053 CSR1Q6 121461772 IC50 > 57000 nM T15053 CV3L8S 121461774 IC50 = 2370 nM T15053 CD38EL 121461780 IC50 > 57000 nM T15053 CDP5S6 121461783 IC50 > 57000 nM T15053 C3DKC7 121461786 IC50 > 57000 nM T15053 C7IX6R 121461805 IC50 = 84 nM T15053 CF8W9O 121461807 IC50 = 110 nM T15053 CMS1Q6 121461818 IC50 = 349 nM T15053 CJG3D2 121461820 IC50 = 9 nM T15053 CW8R2L 121461821 IC50 = 110 nM T15053 CM24KA 121461825 IC50 = 95 nM T15053 C8AC4V 121461896 IC50 = 95 nM T15053 C72VAW 121461897 IC50 = 23400 nM T15053 CV4Z7N 121461900 IC50 = 229 nM T15053 CG24YF 122178659 IC50 = 240 nM T15053 C8KZO2 122178660 IC50 = 2600 nM T15053 CSTB43 122178661 IC50 = 230 nM T15053 CR03XM 122178662 IC50 = 370 nM T15053 CD8HC7 122178663 IC50 = 100 nM T15053 CL63CJ 122178664 IC50 = 170 nM T15053 CP7UV8 122178665 IC50 = 60 nM T15053 C3D2EF 122178666 IC50 = 90 nM T15053 CU4RY3 122178667 IC50 = 100 nM T15053 CWEP16 122178668 IC50 = 60 nM T15053 CY0PR2 122178669 IC50 = 108 nM T15053 CG17IW 122178670 IC50 = 85 nM T15053 C5Z8IF 122178671 IC50 = 1100 nM T15053 CT4VD9 122178672 IC50 = 120 nM T15053 CD72UZ 122178673 IC50 = 370 nM T15053 C8R0OC 122178674 IC50 = 640 nM T15053 C4S1DU 122178675 IC50 = 170 nM T15053 C2BI6T 122178676 IC50 = 3500 nM T15053 CDM80O 122178677 IC50 = 1800 nM T15053 C7N5VJ 122178678 IC50 = 10000 nM T15053 CH0Y2F 122178679 IC50 = 300 nM T15053 C3DYX1 122178680 IC50 = 40 nM T15053 CMOU32 122178681 IC50 = 130 nM T15053 C3G8OB 122178682 IC50 = 120 nM T15053 CU30SE 122178683 IC50 = 90 nM T15053 C1WV6O 122178684 IC50 = 30 nM T15053 CZH21D 122178685 IC50 = 25 nM T15053 C0AN4Z 122178686 IC50 = 15 nM T15053 C7HO8X 122178687 IC50 = 460 nM T15053 CK86PQ 122178688 IC50 = 35 nM T15053 CMF14N 122178689 IC50 = 30 nM T15053 CF36EA 122178690 IC50 = 30 nM T15053 CHNV70 122186806 IC50 = 32000 nM T15053 CS0BR5 122186807 IC50 = 41000 nM T15053 CVO4Q7 122186808 IC50 = 46000 nM T15053 C9T5OB 122186809 IC50 = 41000 nM T15053 C28PGF 122186810 IC50 = 38000 nM T15053 C7ADX5 122186811 IC50 = 115000 nM T15053 C3B8ZU 122186812 IC50 > 200000 nM T15053 C4GHM6 122186813 IC50 > 200000 nM T15053 C83TFK 122187851 IC50 > 200000 nM T15053 COC6P1 122187852 IC50 = 125000 nM T15053 CB5Q3J 127039632 IC50 = 7800 nM T15053 CR70XZ 127041973 Ki = 5460 nM T15053 C07ZRF 127042264 Ki = 1300 nM T15053 C78GJW 127042927 Ki = 3000 nM T15053 CPY46R 127042928 Ki = 200 nM T15053 CUK81P 127042929 Ki = 30 nM T15053 CY65ND 130418263 IC50 > 10000 nM T15053 CMZW49 131801110 IC50 = 55 nM T15053 CCMJ13 131955127 EC50 = 170 nM T15053 C04USK 135335776 IC50 = 25500 nM T15053 CRMN90 135411083 IC50 = 42400 nM T15053 CM2NG5 135415844 IC50 = 12100 nM T15053 CKAF26 135460193 IC50 = 7400 nM T15053 CW09LA 135487739 Ki = 2500 nM T15053 CIDL82 135505406 IC50 > 100000 nM T15053 CP9U1V 135535745 Ki = 600 nM T15053 CCK14U 135667148 IC50 > 100000 nM T15053 C6Q5DF 135667151 IC50 > 100000 nM T15053 CIPZ38 135667152 IC50 = 55700 nM T15053 CQHA97 135667153 IC50 = 50200 nM T15053 C58ALU 135667156 IC50 > 100000 nM T15053 CZ4XA9 135667157 IC50 > 100000 nM T15053 C43KDS 135667161 IC50 = 46800 nM T15053 C20FYS 135667162 IC50 = 26500 nM T15053 CHX49V 135667166 IC50 = 38600 nM T15053 C9KR0Q 135667170 IC50 = 55800 nM T15053 C1G3TN 135667172 IC50 = 22600 nM T15053 C1WH3Z 135891810 IC50 = 8800 nM T15053 CTD83F 135891816 IC50 = 27600 nM T15053 CN0CQ3 136087128 IC50 = 17000 nM T15053 CZ8AB4 136242871 IC50 > 100000 nM T15053 CBO5I1 136242872 IC50 = 480 nM T15053 CQDT25 136242873 IC50 = 750 nM T15053 CK5AZ7 136242878 IC50 = 710 nM T15053 CRU56Z 136242879 IC50 = 650 nM T15053 C9ER5I 137125271 IC50 > 200000 nM T15053 C6W8NF 137631546 IC50 > 57000 nM T15053 CWM2Z3 137634582 IC50 > 57000 nM T15053 CO5DI2 137636531 IC50 = 162 nM T15053 C13BXM 137638998 IC50 = 213 nM T15053 CZT2E6 137639008 IC50 = 1100 nM T15053 C69NZW 137639445 IC50 = 1020 nM T15053 CVH98X 137639861 IC50 = 9570 nM T15053 CDE0M6 137640502 IC50 = 168 nM T15053 C5MZ0T 137641261 IC50 > 57000 nM T15053 CYD4U0 137645277 IC50 = 134 nM T15053 C7Z1LD 137650206 IC50 = 189 nM T15053 C18RXF 137650978 IC50 = 266 nM T15053 CU35MW 137651644 IC50 = 669 nM T15053 CTWD09 137654268 IC50 > 57000 nM T15053 CAC2O0 137655821 IC50 = 299 nM T15053 C9QTP5 137656179 IC50 = 106 nM T15053 CG5HS1 138753630 IC50 > 10000 nM T15053 CJZF96 145966259 IC50 > 500000 nM T15053 C8VF2A 145966736 IC50 > 500000 nM T15053 CDNX87 145969821 IC50 = 102400 nM T15053 C6LW5R 145970499 IC50 > 500000 nM T15053 CAT32J 145971339 IC50 > 500000 nM T15053 CB3F0M 145973103 IC50 > 500000 nM T15053 CDLN05 145976873 IC50 > 500000 nM T15053 CN04BE 145976955 IC50 > 500000 nM T15053 CGN9F5 155510539 IC50 = 21 nM T15053 CMQ36B 155511312 IC50 = 4 nM T15053 CDK81A 155516285 IC50 > 10000 nM T15053 C8UZH1 155516981 IC50 = 42 nM T15053 C1MEF5 155517278 IC50 = 7 nM T15053 CCK7Z2 155518129 IC50 = 100 nM T15053 CIMT08 155520991 EC50 = 1200 nM T15053 CDX9E7 155521878 IC50 = 2900 nM T15053 C95UXN 155523475 IC50 = 15 nM T15053 CK9Z5L 155526375 IC50 > 10000 nM T15053 C0DIQ3 155532490 IC50 = 5 nM T15053 CWRU60 155532931 IC50 = 47 nM T15053 C82XQT 155533013 IC50 = 400 nM T15053 CP8KI3 155536759 IC50 = 80 nM T15053 C67SAM 155537817 IC50 = 10 nM T15053 C5LY1R 155542943 IC50 = 14 nM T15053 C7J3BW 155543065 IC50 = 360 nM T15053 C36FEP 155543547 IC50 = 490 nM T15053 C7R9VA 155545342 IC50 = 700 nM T15053 CESO73 155548785 IC50 = 13 nM T15053 CP8TA9 155549515 IC50 = 3900 nM T15053 CSE6Y5 155552406 IC50 = 15 nM T15053 CATW09 155553170 IC50 = 9 nM T15053 CGU61P 155553810 IC50 = 3 nM T15053 CUT93J 155553855 EC50 = 7500 nM T15053 C9OUQ4 155554510 EC50 = 172000 nM T15053 CR9MK1 155554523 IC50 = 17 nM T15053 CU4KR0 155556866 IC50 = 37 nM T15053 CYA28E 155559570 EC50 = 700 nM T15053 C27QFZ 155562355 IC50 > 10000 nM T15053 CZL7I9 155564050 IC50 = 52 nM T15053 CRO6M5 155565718 IC50 = 58 nM T15053 CF6ML7 155566164 IC50 = 25000 nM T15053 D09ALJ 5280805 IC50 > 500000 nM T15053 D09EDP 448651 IC50 = 54000 nM T15053 D0LP2H 974 Ki = 26000 nM T15053 D0T3PV 448652 IC50 = 10000 nM T45601 C7A9BK 65023 IC50 = 1000 nM T45601 CX0B5L 9853618 IC50 > 100000 nM T45601 C69KGX 10394329 Ki = 8 nM T45601 CW68BJ 11518143 IC50 > 30000 nM T45601 C3LW2D 11632240 IC50 = 29000 nM T45601 CLP92O 11963435 IC50 > 30000 nM T45601 CE29TK 14887165 IC50 = 1000 nM T45601 CJO10Z 14887166 IC50 = 1000 nM T45601 C02NGW 14887167 IC50 = 1000 nM T45601 CJ8R0O 14887174 IC50 = 1000 nM T45601 CHIC86 14887175 IC50 = 1000 nM T45601 C56EWA 14887177 IC50 = 1000 nM T45601 C2LRD8 14887179 IC50 = 1000 nM T45601 CT4V6C 14887181 IC50 = 1000 nM T45601 C4UA0C 14887183 IC50 = 1000 nM T45601 C6JF8N 14887185 IC50 = 1000 nM T45601 CAKS64 14887194 IC50 = 1000 nM T45601 CE12CX 15018069 Ki > 4000 nM T45601 CI41XT 15126555 Ki = 9 nM T45601 CWF5Z3 25143506 IC50 > 30000 nM T45601 CS7XD5 44321765 Ki = 19 nM T45601 C2OFK8 44321766 Ki > 4000 nM T45601 CZ45LH 44322035 Ki > 4000 nM T45601 CQ09YG 44322074 Ki > 4000 nM T45601 C3N9LQ 44322075 Ki > 4000 nM T45601 CK0BQ2 44322083 Ki > 4000 nM T45601 CNT69K 44322084 Ki > 4000 nM T45601 CN58AQ 44322086 Ki = 110 nM T45601 C1G0FY 44322087 Ki > 4000 nM T45601 CMB9W5 44383534 IC50 = 1000 nM T45601 C2PJ4N 59271992 IC50 > 30000 nM T45601 C56CFA 68448803 IC50 > 10000 nM T45601 CS5WE2 90663011 Ki = 9.2 nM T45601 CI5O9G 90663012 Ki = 78 nM T45601 CW3M7K 90663013 Ki = 51 nM T45601 CZG7Q0 90663014 Ki = 7.2 nM T45601 C9CI2T 90663015 Ki = 210 nM T45601 CFVL78 90663019 Ki = 14 nM T45601 C72FWD 91929322 Ki > 4000 nM T45601 D0KK6A 15126552 Ki = 13 nM T45601 D0P6RT 10078814 Ki = 0.9 nM T09770 C8T6GS 13017 Ki = 380000 nM T09770 C6C7ZT 13376 Ki = 30000 nM T09770 CG1I4X 22686 Ki = 21000 nM T09770 CNY4H5 80654 Ki = 11000 nM T09770 CK7LB3 221387 Ki = 180000 nM T09770 CZI0Y4 253317 Ki = 28000 nM T09770 CT83WR 268118 Ki = 210000 nM T09770 C7BCG2 347402 Ki = 740 nM T09770 C6FE8Z 5287890 Ki = 1100000 nM T09770 C0TYR2 10510948 Ki = 4900000 nM T09770 CJR9A3 10535470 Ki = 960000 nM T09770 CP9N5D 10582973 Ki = 1800000 nM T09770 C2OU9B 10654643 Ki = 640000 nM T09770 CI41XN 10654696 Ki = 1300000 nM T09770 CFB7N0 10725554 Ki = 930000 nM T09770 C2HM1K 10773209 Ki = 1700000 nM T09770 CG4Y3W 11815987 Ki = 100000 nM T09770 CA0D9M 15475283 Ki = 300000 nM T09770 CUQ1A8 20333386 Ki = 47000 nM T09770 CZ07CP 20336979 Ki = 54000 nM T56871 D00SUC 74766595 IC50 = 2 nM T56871 D01WHH 90216982 IC50 < 100 nM T56871 D03TKM 76901247 IC50 = 200 nM T56871 D05CCY 77106319 IC50 = 100 nM T56871 D0G8QR 76282772 IC50 < 100 nM T56871 D0GH8J 90204862 IC50 < 100 nM T56871 D0K4LW 90205053 IC50 < 100 nM T56871 CMKP07 736587 IC50 = 1000 nM T56871 CW01ZQ 22581416 IC50 = 29700 nM T56871 CP65KR 22581444 IC50 = 52600 nM T56871 C75LNS 22581449 IC50 = 22700 nM T56871 C4HXD2 76901248 IC50 = 76 nM T56871 C4VGX7 76901615 IC50 = 170 nM T56871 CZC7E1 76901616 IC50 = 500 nM T56871 CC5WE1 76901618 IC50 = 350 nM T56871 CA79XV 76901619 IC50 = 540 nM T56871 CM2L1V 76901620 IC50 = 120 nM T56871 C6IJN1 78426128 IC50 < 1000 nM T56871 CX23ZP 78426670 IC50 = 250 nM T56871 CMR52S 78426698 IC50 = 3 nM T56871 CKXW73 78427224 IC50 < 250 nM T56871 CIG3E9 83672127 IC50 > 100000 nM T56871 CS4Q1F 86268882 IC50 < 100 nM T56871 CRQ51Z 86346639 IC50 < 100 nM T56871 CZ9DC6 86725498 IC50 = 4400 nM T56871 C8WA4M 86725535 IC50 = 1 nM T56871 C8MGN0 86725568 IC50 = 0.6 nM T56871 CT46KN 90094283 IC50 < 1000 nM T56871 CG4BZ9 90094442 IC50 < 100 nM T56871 C9IYE0 90204662 IC50 = 1 nM T56871 CHV05N 90204861 IC50 = 4 nM T56871 C6PI4M 90204893 IC50 = 54 nM T56871 CU8SJ5 90204921 IC50 = 2 nM T56871 C5A3VQ 90204958 IC50 = 8 nM T56871 CIY20E 90204966 IC50 = 6 nM T56871 C6DA2O 90204997 IC50 = 42 nM T56871 CK6L5M 90205111 IC50 = 370 nM T56871 CO8UQ0 90205153 IC50 = 4 nM T56871 C5ST7H 90205231 IC50 = 4 nM T56871 CJ37CO 90205235 IC50 = 100 nM T56871 CQV07L 90205291 IC50 = 3 nM T56871 CJ5E4U 90205326 IC50 = 4 nM T56871 C5W7FL 90205353 IC50 = 1 nM T56871 CR21SC 90205356 IC50 = 230 nM T56871 C7ZVG4 90205376 IC50 = 22 nM T56871 CM2NA1 90205425 IC50 = 4 nM T56871 CB7Z0A 90205426 IC50 = 4 nM T56871 CN9I0J 90205512 IC50 = 240 nM T56871 C2T4RD 90205719 IC50 = 24 nM T56871 C9H8PV 90211058 IC50 = 41 nM T56871 C1GBT5 90225370 IC50 < 100 nM T56871 CFX8E0 90407594 IC50 = 100 nM T56871 CJ9OZ4 90407809 IC50 = 100 nM T56871 C5LDR2 90407841 IC50 < 100 nM T56871 C7MXT5 90454779 EC50 = 530 nM T56871 CQY0K3 91938043 IC50 < 250 nM T56871 CP3DK0 96607511 IC50 = 12 nM T56871 C85UGZ 96608360 IC50 = 1300 nM T56871 CCZ4Q9 96617507 IC50 = 98 nM T56871 CY87WL 112499933 IC50 = 2200 nM T56871 CT04PB 118420691 IC50 < 250 nM T56871 CPSD31 118420829 IC50 < 250 nM T56871 CJSP15 118420859 IC50 < 250 nM T56871 CU94QR 118421047 IC50 < 250 nM T56871 CH6FX3 118421371 IC50 < 250 nM T56871 C6YT2Q 118598059 IC50 = 750 nM T56871 C7TBE9 118908379 IC50 = 4.7 nM T56871 CJVK69 119081409 IC50 = 56 nM T56871 CRM93S 122181583 IC50 = 9240 nM T56871 CIJ0G6 127030272 IC50 < 250 nM T56871 CN16WB 127030937 IC50 < 100 nM T56871 C2FPM6 127031758 IC50 = 590 nM T56871 C7W8TS 127031759 IC50 = 40 nM T56871 CMJE83 127031760 IC50 = 130 nM T56871 CDC17F 127032730 IC50 = 1000 nM T56871 CL38FP 127033048 IC50 < 100 nM T56871 C2EY1K 127033166 IC50 < 250 nM T56871 CID1E9 127034046 IC50 < 250 nM T56871 CT4O5U 135567037 IC50 = 12000 nM T56871 CC4H1N 135567038 IC50 = 2700 nM T56871 CQBH95 135567040 IC50 = 72000 nM T56871 CP6IH9 135567041 IC50 = 19000 nM T56871 C8HMG2 135567042 IC50 = 22000 nM T56871 C2Z6CV 135567105 IC50 = 124 nM T56871 CIW61V 135567106 IC50 = 1300 nM T56871 CNZ8K9 135567107 IC50 = 310 nM T56871 CL9ZD4 135567108 IC50 = 42 nM T56871 CJM4Z2 135567109 IC50 = 350 nM T56871 CDY98J 135567110 IC50 = 30 nM T56871 C1VAI3 135567112 IC50 = 14 nM T56871 CWI0N7 135567114 IC50 = 7000 nM T56871 C8LFY7 135567115 IC50 = 14 nM T56871 C5E0ZN 135567116 IC50 = 690 nM T56871 CWCY64 136048725 IC50 = 4600 nM T56871 CT0DW5 136048747 IC50 < 100 nM T56871 CXW0S7 136048748 IC50 < 100 nM T56871 CJ91RY 136048749 IC50 < 100 nM T56871 CU10SL 136258480 IC50 = 320 nM T56871 C1H9NK 136959977 IC50 < 100 nM T56871 CF5XJ1 137146154 IC50 = 4100 nM T56871 CK8DR7 137174994 IC50 = 71 nM T56871 CA6DH2 137174995 IC50 = 199 nM T56871 CLDH80 137174999 IC50 = 48 nM T56871 CR37AY 137175000 IC50 = 72 nM T56871 C1J3YB 137175001 IC50 = 48 nM T56871 CGAS95 137175002 IC50 = 48 nM T56871 CS5C6F 137175084 IC50 = 21400 nM T56871 C7PZ2T 137175085 IC50 = 630 nM T56871 C1B5CK 137175086 IC50 = 1400 nM T56871 CWV4Y6 137175087 IC50 = 3900 nM T56871 C9XOV5 137175088 IC50 = 2000 nM T56871 C34LUV 137175094 Ki = 2 nM T56871 CSWN28 137175120 IC50 = 43 nM T56871 C23GYQ 137175121 IC50 = 11 nM T56871 C8Y2PR 137175122 IC50 = 18 nM T56871 C7GUC3 137175140 IC50 = 16 nM T56871 CBD1Q8 137175175 IC50 = 26 nM T56871 CEL6B1 137175176 IC50 = 43 nM T56871 C7SC6T 137175177 IC50 = 18 nM T56871 CPU73A 137175178 IC50 = 10 nM T56871 CFJ76N 137175179 IC50 = 56 nM T56871 CA89LW 137175180 IC50 = 58 nM T56871 C5GV3Q 137175209 IC50 = 15 nM T56871 C93YUK 137175210 IC50 = 26 nM T56871 CB2XV7 137175225 IC50 = 66000 nM T56871 C0XN8Y 137175239 IC50 = 7000 nM T56871 CI4D3P 137175249 IC50 = 21 nM T56871 CTVD83 137175250 IC50 = 17 nM T56871 C80LCT 137175251 IC50 = 15 nM T56871 CKQ1I2 137175252 IC50 = 15 nM T56871 C1YGB9 137175253 IC50 = 28 nM T56871 C5OZR6 137175260 IC50 = 10 nM T56871 CIKW02 137175261 IC50 = 7 nM T56871 C7J1RC 138393333 IC50 = 156 nM T56871 CYG29R 138393334 Ki = 4 nM T56871 CNG82D 138393336 Ki = 7 nM T56871 CPFZ83 138393339 IC50 = 68 nM T56871 CC6SU2 138393341 Ki = 2 nM T56871 C1ANF3 138518187 IC50 = 70 nM T56871 CXV31U 138753208 IC50 = 80 nM T56871 C41KVR 138753209 IC50 = 26 nM T56871 CIQJ26 138753211 Ki = 1 nM T56871 CARJ34 138753212 Ki = 16 nM T56871 CEQD63 155510449 IC50 = 32 nM T56871 CCB54Y 155510907 IC50 = 114 nM T56871 CAMR98 155512849 IC50 = 127 nM T56871 C9TWS3 155514456 IC50 = 12 nM T56871 C7XNM9 155518054 IC50 = 601 nM T56871 C4M1EO 155519111 Ki = 3 nM T56871 CRT5Z2 155525082 IC50 = 439 nM T56871 CMB9N3 155530704 IC50 = 123 nM T56871 C2HN9G 155536799 IC50 = 66 nM T56871 C7VX3Y 155538517 IC50 = 51 nM T56871 CP8K5E 155540290 IC50 = 17 nM T56871 C7LFH3 155540572 IC50 = 131 nM T56871 CTF1K9 155542268 IC50 = 25 nM T56871 C7EG9J 155543678 IC50 = 81 nM T56871 C3M0TR 155546359 IC50 = 447 nM T56871 CIM7D4 155548682 IC50 = 51.1 nM T56871 C1CNK5 155549007 IC50 = 23 nM T56871 CX9OP1 155550806 IC50 = 48 nM T56871 CFR06L 155551969 IC50 = 1.34 nM T56871 C48ANL 155557731 IC50 = 21 nM T56871 C4MU5J 155558505 IC50 = 149 nM T56871 CTDM51 155558717 IC50 = 42 nM T56871 CPOM30 155560356 Ki = 1 nM T56871 CA9T8I 155563296 IC50 = 146 nM T56871 CGCN43 155567831 IC50 = 41 nM T56871 C3SQ4A 155569285 IC50 = 12 nM T56871 D07IOY 10365 IC50 = 2700 nM T56871 D0P7MU 4119262 IC50 = 51200 nM T15739 D0W7HE 56649450 IC50 > 10000 nM T15739 C14ONZ 8822251 EC50 = 12 nM T15739 CDAT72 11433190 IC50 = 1000 nM T15739 C37TYU 18125907 EC50 = 9 nM T15739 C42VTB 35972429 EC50 = 4 nM T15739 CO7Y2Z 44519134 EC50 = 80 nM T15739 C06PGX 45483723 IC50 = 1000 nM T15739 CI9B2K 45483728 IC50 = 6500 nM T15739 C09ZQE 45483731 IC50 = 44300 nM T15739 CCKD24 45483751 IC50 = 9370 nM T15739 CVJ6E9 45483794 IC50 = 15000 nM T15739 CT5GN4 45483803 IC50 = 11400 nM T15739 CCSL17 56591137 IC50 = 5500 nM T15739 CYH8K7 56591154 IC50 = 1000 nM T15739 CW78DN 56591304 IC50 = 10700 nM T15739 CG0R8H 56591324 IC50 = 4300 nM T15739 CQ8Y7H 56591370 IC50 = 34400 nM T15739 C15HTM 56965957 IC50 = 760 nM T15739 C59YAC 57495353 IC50 > 3000 nM T15739 CE5R2U 58573876 IC50 = 1500 nM T15739 C7FZ8S 60154126 IC50 = 3100 nM T15739 C3VJG9 67998380 IC50 = 1600 nM T15739 CQ57FD 89699436 EC50 = 65 nM T15739 CCND47 89699460 EC50 = 74 nM T15739 C2KQ3B 89699467 EC50 = 152 nM T15739 CP23ZQ 89699521 EC50 = 2 nM T15739 C5DJ2T 89699688 EC50 = 158 nM T15739 C3SF4B 101911084 IC50 = 6200 nM T15739 CR9ND4 118735492 IC50 = 6200 nM T15739 C68XSE 145982731 EC50 = 4 nM T15739 CT7Z9D 145985742 EC50 > 5000 nM T15739 D00DXI 135566302 IC50 = 5000 nM T15739 D03XXT 72201027 IC50 = 1540 nM T15509 D0T9TJ 3034010 IC50 = 60 nM T15509 CC3Y8W 45040160 IC50 = 25.12 nM T15509 C8PJ6E 53354789 IC50 = 40 nM T15509 CXS23L 53373470 IC50 = 146 nM T15509 CT6K2O 53373472 IC50 = 112 nM T15509 C1LOV9 53373473 IC50 = 80 nM T15509 CHT12Z 127039880 IC50 = 40 nM T15509 CI3L5S 155534105 IC50 = 6.31 nM T15509 D05LXG 5063 IC50 = 60 nM T03878 C4V2NK 145965586 IC50 = 254000 nM T03878 C6SU5D 145977503 IC50 = 1300 nM T03878 C9X4RK 154702459 IC50 = 396 nM T03878 C1K0TP 154702460 IC50 = 206 nM T03878 C6YI0M 154702461 IC50 > 250000 nM T03878 CL0R4A 154702462 IC50 > 250000 nM T96079 D0L5RW 65015 IC50 = 0.057 ug.mL-1 T96079 D0Z9QR 24066 EC50 = 88 nM T96079 D00XBC 46861584 IC50 > 10000 nM T96079 D0O2XQ 11256587 IC50 = 13 nM T96079 D0G6SZ 3001322 IC50 = 30000 nM T96079 C92TML 65014 IC50 = 12.4 nM T96079 CK04YH 203317 IC50 > 10000 nM T96079 CTL81I 248372 EC50 = 1000000 nM T96079 CQX4M9 265219 IC50 > 60000 nM T96079 CHOP34 460326 IC50 = 67 nM T96079 CQFL73 460344 Ki = 2300 nM T96079 C0OM4E 465968 IC50 = 13 nM T96079 CGYT63 477101 IC50 = 5737 nM T96079 CQN85D 477103 IC50 > 35000 nM T96079 CEB52A 477104 IC50 = 1 nM T96079 C2ORC4 477106 IC50 = 4363 nM T96079 C23LNG 478459 IC50 > 35000 nM T96079 CHNV85 478460 IC50 > 35000 nM T96079 CR7A3C 478462 IC50 > 35000 nM T96079 CYUP05 478464 IC50 > 35000 nM T96079 CQ3KO7 483339 IC50 > 1000 nM T96079 C7AP9W 483340 IC50 > 1000 nM T96079 CAB79M 483341 IC50 > 1000 nM T96079 C7XW2D 483342 IC50 > 1000 nM T96079 C7PMT6 483343 IC50 > 1000 nM T96079 CP25RI 483344 IC50 > 1000 nM T96079 CN78FW 483559 Ki = 10 nM T96079 CLH45E 483570 Ki = 170 nM T96079 CA5BZ8 491773 IC50 = 6700 nM T96079 CB27WS 849733 IC50 > 10000 nM T96079 CT6OG0 1259151 IC50 > 10000 nM T96079 C78UJK 2236109 IC50 = 10000 nM T96079 CPB2J9 2795811 IC50 = 3800 nM T96079 CQNJ07 3313778 EC50 = 100000000 nM T96079 COT07B 3453336 IC50 > 60000 nM T96079 CNH6R0 4225968 EC50 = 1000000 nM T96079 CO5F3T 4294941 EC50 = 39810717.06 nM T96079 CB0Y3Z 4719657 IC50 > 10000 nM T96079 CH5M7D 5218952 EC50 = 1000000 nM T96079 C13TYG 5275846 IC50 = 180 nM T96079 CY0G8T 5275847 IC50 = 32 nM T96079 C6NMB2 5275848 IC50 = 190 nM T96079 C0C6LX 5278944 IC50 = 1000 nM T96079 C7YO6C 5278945 IC50 = 530 nM T96079 CPKQ82 5278946 IC50 = 1000 nM T96079 CEMG40 5278947 IC50 > 10000 nM T96079 CQ4L7V 5278948 IC50 > 10000 nM T96079 CBX93L 5278953 IC50 = 4.3 nM T96079 CRA02D 5278955 IC50 = 420 nM T96079 CS12MC 5278956 IC50 = 1600 nM T96079 CD2BE1 5278957 IC50 = 63 nM T96079 CSXV96 5278958 IC50 = 490 nM T96079 CX60AF 5278959 IC50 = 230 nM T96079 C2EK9M 5278960 IC50 = 42 nM T96079 C02KHJ 5278961 IC50 = 16 nM T96079 C5VR9W 5278962 IC50 = 19 nM T96079 C0C1RU 5278963 IC50 = 97 nM T96079 C3MR9Q 5278964 IC50 = 24 nM T96079 C4L5DQ 5278965 IC50 = 33 nM T96079 CK8WF2 5278969 IC50 = 10 nM T96079 C8AE4V 5278970 IC50 = 9.9 nM T96079 CL45FU 5708903 Ki = 53 nM T96079 C65VZI 5943987 IC50 = 2160 nM T96079 C81BDY 8241537 EC50 = 100000000 nM T96079 CX04VC 8241714 EC50 = 1000000000 nM T96079 CO5D1L 9887073 IC50 = 1402 nM T96079 CSH40U 9936494 IC50 > 10000 nM T96079 C62OTD 9959718 IC50 = 250 nM T96079 C2U0SM 10010259 IC50 = 290 nM T96079 C5TWF9 10055825 IC50 = 2200 nM T96079 CWF87Z 10078747 IC50 = 23000 nM T96079 C49DEF 10117347 IC50 > 30000 nM T96079 CH7KZ9 10126019 IC50 = 11 nM T96079 C9NDC8 10149770 IC50 = 1369 nM T96079 C2U4WP 10159217 IC50 > 30000 nM T96079 CS5Y9X 10172242 IC50 = 160 nM T96079 C1BGH8 10182763 IC50 > 30000 nM T96079 C2ED3X 10184169 IC50 > 10000 nM T96079 C6KC3U 10198583 IC50 = 200 nM T96079 CXK43P 10204589 IC50 > 30000 nM T96079 C4OM2Z 10205915 IC50 > 10000 nM T96079 CWC7X1 10208080 IC50 > 10000 nM T96079 C0NID4 10215423 IC50 = 973 nM T96079 C72HMR 10228761 IC50 > 30000 nM T96079 CWU1V9 10237323 IC50 = 87 nM T96079 C3CZ7H 10277466 IC50 > 10000 nM T96079 CE9ID0 10280944 IC50 > 10000 nM T96079 C04WUS 10286987 IC50 = 190 nM T96079 CO0P4F 10301330 IC50 > 10000 nM T96079 C3OKR9 10308735 IC50 = 68 nM T96079 CPH6M3 10372866 IC50 = 2 nM T96079 CR2J6L 10485171 IC50 = 6000 nM T96079 C74XEH 10502669 IC50 > 7 nM T96079 C3PBD8 10740531 IC50 > 7 nM T96079 C9X7DQ 11233382 IC50 = 206 nM T96079 C1NP4I 11310349 IC50 > 10000 nM T96079 C8FT3O 11411355 IC50 = 690 nM T96079 C9F6ZX 11489510 IC50 < 4 nM T96079 C4FI3V 11505556 EC50 = 51000 nM T96079 CG1KV3 11565518 EC50 = 0.3 nM T96079 C1DKF4 11598797 IC50 > 10000 nM T96079 CPAY69 11625279 IC50 = 76 nM T96079 C57RHQ 11634966 IC50 > 10000 nM T96079 C4MB0X 11635914 IC50 > 1000 nM T96079 C57VGY 11638842 IC50 = 47 nM T96079 C6MOD0 11648393 IC50 = 27 nM T96079 CJEQ78 11678324 IC50 = 11 nM T96079 C04LUA 11686297 IC50 = 51 nM T96079 C1CV9H 11706779 IC50 < 4 nM T96079 C7OWM0 11950261 IC50 = 0.61 nM T96079 COG3X8 14847939 EC50 = 5011872.34 nM T96079 CBP3Z2 15604176 IC50 < 20 nM T96079 CTU1P4 15604290 IC50 < 20 nM T96079 C70MXQ 15959068 IC50 = 4.5 nM T96079 CMPQ63 16102648 IC50 > 30000 nM T96079 C0UZN8 16102649 IC50 > 30000 nM T96079 CWQ03V 16102650 IC50 > 30000 nM T96079 C0EKY9 16102652 IC50 > 30000 nM T96079 CD51PH 16102653 IC50 > 30000 nM T96079 CV59GK 16459886 IC50 = 10000 nM T96079 CU2S9J 16727404 IC50 = 7 nM T96079 CEWL01 17221518 IC50 > 10000 nM T96079 CR2V5A 18665182 IC50 > 7 nM T96079 CN7R4T 20725627 IC50 = 39 nM T96079 C7OMJ8 21984983 IC50 = 28 nM T96079 CD5EX6 21984993 IC50 = 219 nM T96079 CHZ0J3 21984997 IC50 = 126 nM T96079 C9Q1FH 21985008 IC50 = 119 nM T96079 C12EUA 21985015 IC50 = 15 nM T96079 CBM97D 21985038 IC50 = 10 nM T96079 C28KJB 21985074 IC50 = 11 nM T96079 CS1N0Q 21985109 IC50 = 21 nM T96079 CI4SW1 21985119 IC50 = 160 nM T96079 C15SBD 21985149 IC50 = 51 nM T96079 C5MNZ7 22163152 EC50 = 19952623.15 nM T96079 C2Y4HF 22940860 IC50 > 7 nM T96079 COV20C 23653628 IC50 = 5.4 nM T96079 CXPW53 23656445 EC50 = 100000000 nM T96079 C2W7KR 23656597 EC50 = 1000000000 nM T96079 CW4ZH3 23656762 EC50 = 1000000 nM T96079 C1OU6L 23656763 EC50 = 10000000 nM T96079 C51GKY 23656764 EC50 = 1000000000 nM T96079 CT8K9L 24274895 IC50 > 10000 nM T96079 C79SUY 24894090 IC50 = 1200 nM T96079 CV7S9D 25050377 IC50 < 1000 nM T96079 CT4YG7 25177627 IC50 = 44 nM T96079 C8N4XG 25177628 IC50 = 23 nM T96079 CYGQ46 25177629 IC50 = 66 nM T96079 CQYW25 25177630 IC50 = 183 nM T96079 C8M2CQ 25177631 IC50 = 20 nM T96079 C7XRO8 25177632 IC50 = 72 nM T96079 CE9YT1 25178134 IC50 = 3835 nM T96079 CRI46D 25178136 IC50 = 25 nM T96079 C57CRY 25178138 IC50 = 6.6 nM T96079 C5YNR1 25178140 IC50 = 173 nM T96079 C9YCZ1 25178142 IC50 = 304 nM T96079 C51ONB 25178144 IC50 = 13 nM T96079 CR4F6L 25178347 IC50 = 5275 nM T96079 CHTN25 25178350 IC50 = 8120 nM T96079 C4QLV8 25178353 IC50 = 8.8 nM T96079 C5GL9B 25178561 IC50 > 10000 nM T96079 CL5ED0 25178563 IC50 = 5.3 nM T96079 CC3ZM5 25178565 IC50 = 8 nM T96079 C3WI8C 25178567 IC50 = 75 nM T96079 CZ4U9H 25178569 IC50 = 1533 nM T96079 CSI4V6 25178764 IC50 = 9130 nM T96079 C8L4JB 25178766 IC50 = 57 nM T96079 C9P8IV 25181075 IC50 = 931 nM T96079 C54LQF 25230828 IC50 > 50000 nM T96079 C8L1KG 43130924 IC50 > 10000 nM T96079 CI50RO 44400178 IC50 = 10000 nM T96079 CDBO95 44400179 IC50 = 10000 nM T96079 C95AIV 44400199 IC50 = 97 nM T96079 CPLC40 44400262 IC50 = 270 nM T96079 C6LT7U 44400263 IC50 = 170 nM T96079 C1MC8Q 44400264 IC50 = 610 nM T96079 C2DWT3 44400298 IC50 = 54 nM T96079 CE38CQ 44400299 IC50 > 1000 nM T96079 CK51EI 44400300 IC50 > 1000 nM T96079 CW5UM2 44400301 IC50 > 1000 nM T96079 C8K0HX 44400314 IC50 = 10000 nM T96079 CFL7M8 44400315 IC50 = 10000 nM T96079 CH9N5Y 44400758 IC50 = 4.5 nM T96079 CIA5W4 44400868 IC50 > 100000 nM T96079 CN1W7Y 44418864 IC50 > 1000 nM T96079 CVRH73 44418866 IC50 > 1000 nM T96079 C7IV9P 44418867 IC50 > 1000 nM T96079 C4VW8Z 44418870 IC50 > 1000 nM T96079 CB6PG2 44418871 IC50 > 1000 nM T96079 C7V5QA 44418874 IC50 > 1000 nM T96079 CHS01L 44418875 IC50 > 1000 nM T96079 CMU4R9 44418876 IC50 > 1000 nM T96079 C90MUE 44418877 IC50 > 1000 nM T96079 CW3Y8F 44418881 IC50 > 1000 nM T96079 C6KLE2 44418882 IC50 > 1000 nM T96079 CTEF64 44418884 IC50 > 1000 nM T96079 CGA5R6 44435744 EC50 = 5011872.34 nM T96079 CT5N4E 44555481 IC50 > 50000 nM T96079 C6Z9KH 44561446 IC50 = 3000 nM T96079 C6Z9DN 44561483 IC50 = 3000 nM T96079 C1GZ7N 44561487 IC50 = 4800 nM T96079 CPW0H4 44561524 IC50 = 2700 nM T96079 C1V8NG 44561525 IC50 = 2200 nM T96079 CMJ89P 44561526 IC50 = 1700 nM T96079 C6AL9F 44561527 IC50 = 3700 nM T96079 CNUG76 44563599 IC50 = 109 nM T96079 C0F9WE 44563689 IC50 = 2220 nM T96079 C9NLA7 45182189 EC50 = 1900 nM T96079 CJ5QF4 46189876 IC50 = 400 nM T96079 C15WHG 46204208 IC50 = 77 nM T96079 C18GHV 46204209 IC50 = 514 nM T96079 CY1J2K 46204210 IC50 = 75 nM T96079 CF0T4H 46204212 IC50 = 3200 nM T96079 C68YLT 46206136 IC50 = 29200 nM T96079 CK3N1G 46206137 IC50 = 120 nM T96079 CG5EA4 46222002 IC50 = 8.59 ug.mL-1 T96079 CK8QW4 46225413 IC50 > 60000 nM T96079 CSOB03 46830205 IC50 = 3.4 nM T96079 CH96GT 46871630 IC50 = 1.21 ug.mL-1 T96079 C9KJG4 46884785 IC50 = 442 nM T96079 C7DJF1 46888654 IC50 = 74 nM T96079 CC6L0Q 46888759 IC50 = 16 nM T96079 CWV58S 49857283 IC50 = 0.8 nM T96079 CL65OY 50942117 IC50 = 19.8 nM T96079 CQE6Y5 50942118 IC50 = 44.5 nM T96079 CT97QO 51031036 IC50 = 8.9 nM T96079 CRY27T 51346842 IC50 = 62.9 nM T96079 CK95IC 51346844 IC50 = 96.1 nM T96079 CN35PV 51346852 IC50 = 10.9 nM T96079 C4ITX3 52945203 EC50 = 5.9 nM T96079 CZ5WX0 53316607 IC50 = 5 nM T96079 C3AP8D 53318414 IC50 = 49 nM T96079 C18PAS 53319240 IC50 = 60 nM T96079 CDH84L 53319745 IC50 = 91 nM T96079 CE34ZN 53319746 IC50 = 63 nM T96079 CZ1LS0 53320374 IC50 = 5 nM T96079 C7RUM3 53320547 IC50 = 88.9 nM T96079 C8CIN4 53321037 IC50 = 35 nM T96079 C1KQ9G 53321038 IC50 = 38 nM T96079 CX82CB 53321039 IC50 = 19 nM T96079 CWX61J 53321040 IC50 = 27 nM T96079 CHS6Z9 53321041 IC50 = 79 nM T96079 C5NGJ4 53321478 IC50 = 35.8 nM T96079 CJU85F 53321859 IC50 = 21 nM T96079 CKZQ31 53322384 IC50 = 18 nM T96079 CJ4Z7B 53322385 IC50 = 53 nM T96079 C68ZWH 53322799 IC50 = 18 nM T96079 CO45XU 53322803 IC50 = 16.6 nM T96079 C35CGN 53323182 IC50 = 1.3 nM T96079 CW2K4R 53323183 IC50 = 21 nM T96079 C69EAG 53324117 IC50 = 25 nM T96079 C14HXE 53324136 IC50 = 8 nM T96079 C89OYV 53325426 IC50 = 12 nM T96079 CW0V7O 53325442 IC50 = 111 nM T96079 CGU98X 53326307 IC50 = 1621 nM T96079 CPQG17 53326308 IC50 = 129 nM T96079 C3S4EA 53326939 IC50 = 13 nM T96079 CE02UZ 53344611 IC50 = 4.2 nM T96079 CQCT85 53344613 IC50 = 16 nM T96079 CUQ71L 56647829 IC50 = 67 nM T96079 C0S4JM 56649212 IC50 = 1000 nM T96079 C1DOB2 56649213 IC50 = 60 nM T96079 CHM6Z8 56750906 IC50 = 10000 nM T96079 CO4U8S 56955853 IC50 = 36.2 nM T96079 CP7KM4 57343752 IC50 = 6 nM T96079 CL6XH2 57343753 IC50 = 2 nM T96079 CAS5J4 57343965 IC50 = 250 nM T96079 CX9A5N 57343966 IC50 > 30000 nM T96079 C0S1BR 57343967 IC50 > 30000 nM T96079 C1UM9E 57345319 IC50 = 1360 nM T96079 CL45WN 57345320 IC50 = 6 nM T96079 CA7LH0 57345321 IC50 = 190 nM T96079 C9TCP0 57345322 IC50 = 230 nM T96079 C0I3ZR 57400274 IC50 = 6 nM T96079 CDP72K 59826001 IC50 = 8 nM T96079 CIR29B 66545960 IC50 = 9.4 nM T96079 C9O5CX 66558669 IC50 = 679 nM T96079 CE0OV5 66558750 IC50 = 11 nM T96079 CCA09Q 66902958 IC50 = 150 nM T96079 CKL32M 67501386 IC50 = 15 nM T96079 CLAW03 70681869 IC50 = 4.9 nM T96079 CK5T1W 70685748 IC50 > 10000 nM T96079 C7H3UT 70694123 IC50 = 330 nM T96079 CG0VL2 70694124 IC50 = 2500 nM T96079 CX7R6W 70694125 IC50 = 100 nM T96079 CU2O4K 70694478 IC50 = 334 nM T96079 C3XMN4 70694810 IC50 = 0.5 nM T96079 C9EV2G 70695561 IC50 = 31000 nM T96079 CKTD54 70696255 IC50 = 500 nM T96079 CED12U 70887092 IC50 = 800 nM T96079 CG47KL 70887095 IC50 = 600 nM T96079 CCT1Q2 70887131 IC50 = 600 nM T96079 C3G7BP 71450125 IC50 = 1.84 ug.mL-1 T96079 CTE2J1 71450127 IC50 = 1.1 ug.mL-1 T96079 CF2A5N 71450139 EC50 > 100000 nM T96079 CF3A0H 71450175 EC50 = 560 nM T96079 C6SDI0 71450913 IC50 = 21000 nM T96079 CI1OL6 71451639 IC50 = 350 nM T96079 C5SY8N 71451966 EC50 = 14791.08 nM T96079 C2Y1UE 71451968 EC50 = 2884.03 nM T96079 C8UDI9 71452002 EC50 = 257.04 nM T96079 CVS14E 71453764 IC50 = 2.05 ug.mL-1 T96079 CV9I6A 71453766 IC50 = 1.91 ug.mL-1 T96079 CIRV35 71455186 IC50 = 1100 nM T96079 CXZ3N8 71455540 EC50 = 3548.13 nM T96079 CFM9C7 71455543 EC50 = 7200 nM T96079 CLO4B6 71456969 IC50 = 790 nM T96079 CUJ52B 71457283 IC50 = 1.27 ug.mL-1 T96079 CT8GF5 71457301 EC50 = 676.08 nM T96079 C0XN6O 71459134 EC50 < 100000 nM T96079 COQ1L0 71462701 EC50 = 36000 nM T96079 CK7F4J 71462703 EC50 = 5370.32 nM T96079 CSGJ08 71589166 IC50 = 260 nM T96079 CL3F8Y 71589167 IC50 = 280 nM T96079 CSP87Z 71589203 IC50 = 510 nM T96079 C7A4YC 71590315 IC50 = 200 nM T96079 C3FLC2 71590395 IC50 = 680 nM T96079 C9DQP7 71680586 IC50 = 40 nM T96079 CD17OI 71716524 IC50 = 220 nM T96079 C9TWE8 71716525 IC50 = 110 nM T96079 CA2PM9 71716526 IC50 = 300 nM T96079 C3PAX7 71718363 IC50 = 190 nM T96079 C7EQB8 71718364 IC50 = 110 nM T96079 CAG5X2 71718960 IC50 = 180 nM T96079 CNOE61 71719569 IC50 = 93 nM T96079 C7IRO4 71719570 IC50 = 380 nM T96079 C47MEW 71720811 IC50 = 62 nM T96079 CRF0N4 72545830 IC50 = 56 nM T96079 C9KM0Z 72546061 IC50 = 70 nM T96079 C5J8WE 72546062 IC50 = 60 nM T96079 CGL64Q 72546063 IC50 = 490 nM T96079 C7YJ4F 72546064 IC50 = 80 nM T96079 CB32VZ 72546065 IC50 = 20 nM T96079 CDB7W4 72546066 IC50 = 20 nM T96079 C0RY9E 72546294 IC50 = 8 nM T96079 CDW8I1 72546295 IC50 = 7 nM T96079 CM58AK 72736896 EC50 = 31000 nM T96079 CJZX20 72736898 EC50 = 29000 nM T96079 COI0G7 72736900 EC50 = 19000 nM T96079 CW96KP 72737063 EC50 = 5600 nM T96079 CFT12G 72737246 EC50 = 25000 nM T96079 CXJ7F2 72737615 EC50 = 5100 nM T96079 C3C5TA 73345441 EC50 = 2.8 nM T96079 CSYC75 73345442 EC50 = 880 nM T96079 CPWG74 73345443 EC50 = 3.3 nM T96079 C1H2LA 73345746 EC50 = 37 nM T96079 CX4FU8 73346966 EC50 = 15 nM T96079 CZID04 73346967 EC50 = 15 nM T96079 C0FOT5 73346968 EC50 = 16 nM T96079 CQ2KI7 73346969 EC50 = 16 nM T96079 CEY5W7 73347229 EC50 = 40 nM T96079 C7YU4K 73348196 EC50 = 56 nM T96079 C6LRK1 73348466 EC50 = 4 nM T96079 C0A1ST 73348745 EC50 = 6.6 nM T96079 CZ24AH 73348746 EC50 = 4.6 nM T96079 COTU03 73350048 EC50 = 17 nM T96079 CJZ05F 73350052 EC50 = 1300 nM T96079 CH9DQ3 73350053 EC50 = 2500 nM T96079 CQWH52 73350054 EC50 = 9.3 nM T96079 CYQZ02 73350055 EC50 = 17 nM T96079 C1DVR5 73350320 EC50 = 0.6 nM T96079 C3G2BN 73351279 EC50 = 400 nM T96079 C36WVS 73351552 EC50 = 8.3 nM T96079 CPMY91 73351833 EC50 = 68 nM T96079 CTZ5F6 73351834 EC50 = 8.9 nM T96079 C2KRH1 73351835 EC50 = 0.5 nM T96079 CZWL45 73353307 EC50 = 3.3 nM T96079 C4N6TK 73353309 EC50 = 2.7 nM T96079 C59UVE 73353310 EC50 = 4 nM T96079 C75LDY 73353311 EC50 = 6.8 nM T96079 CR80IC 73353312 EC50 = 1.2 nM T96079 C93EGT 73354527 EC50 = 47 nM T96079 C35SVZ 73354528 EC50 = 450 nM T96079 CJ06OA 73354530 EC50 = 16 nM T96079 C9XH6U 73354822 EC50 = 7.8 nM T96079 C04SOR 73354823 EC50 = 2.8 nM T96079 CU3B4H 73354824 EC50 = 36 nM T96079 CM9XS2 73356099 EC50 = 360 nM T96079 CVJ20Q 73356100 EC50 = 18 nM T96079 CPQ6Z5 73356370 EC50 = 0.4 nM T96079 CMSL68 73356371 EC50 = 72 nM T96079 C0RE7B 76309931 IC50 = 180 nM T96079 CXW94C 76313651 IC50 = 450 nM T96079 CR7FP8 76324529 IC50 = 1 nM T96079 CCY51M 76331766 IC50 = 210 nM T96079 CL20JG 76335355 IC50 = 4 nM T96079 C6ENV5 100951623 EC50 > 10000 nM T96079 C07SEY 118712250 EC50 = 57543.99 nM T96079 CN5S0D 118712251 EC50 = 85113.8 nM T96079 C6YL3G 118712252 EC50 = 43651.58 nM T96079 CNZB65 118712253 EC50 < 100000 nM T96079 CSF68W 118712254 EC50 < 100000 nM T96079 C6YK0F 118712255 EC50 < 100000 nM T96079 C2IY3M 118712256 EC50 < 100000 nM T96079 C2Y3NX 118712257 EC50 = 60000 nM T96079 CC5D7O 118712258 EC50 > 100000 nM T96079 C34JVT 118712259 EC50 > 100000 nM T96079 CQ8JX0 118712260 EC50 = 79432.82 nM T96079 C7O0JI 118712261 EC50 = 63095.73 nM T96079 C2TH7D 118722241 IC50 = 15100 nM T96079 CJY36P 118724116 IC50 = 5.2 nM T96079 CCX93Y 118724117 IC50 = 6.7 nM T96079 CEF53C 118965334 IC50 = 34.1 nM T96079 CV12LX 118965366 IC50 = 71.1 nM T96079 C9LR8Z 118965395 EC50 = 13.7 nM T96079 C0VSJ9 118965398 IC50 = 97.6 nM T96079 CJ6HV4 118965421 IC50 = 158 nM T96079 CNUO35 118965426 IC50 = 93 nM T96079 C6CTB8 121595992 IC50 = 53 nM T96079 CNO35Z 121595994 IC50 = 53 nM T96079 C7W0LF 122178716 IC50 > 30000 nM T96079 CQ4Y2B 122178717 IC50 = 4600 nM T96079 C4X5HK 122178718 IC50 > 30000 nM T96079 CX0D2P 122178719 IC50 > 30000 nM T96079 CXJ01F 122178720 IC50 > 30000 nM T96079 CCZF85 122178721 IC50 > 30000 nM T96079 C1HM2J 122178722 IC50 > 30000 nM T96079 CJ5FP0 122178723 IC50 > 30000 nM T96079 C5NT4D 122178724 IC50 > 30000 nM T96079 CR8AJ9 122178725 IC50 > 30000 nM T96079 CM6W9J 122178726 IC50 > 30000 nM T96079 CE1AR2 122178727 IC50 > 30000 nM T96079 CV7UY5 122178728 IC50 > 30000 nM T96079 C8EJT2 122178729 IC50 > 30000 nM T96079 CN6S8D 122178730 IC50 > 30000 nM T96079 C19BRQ 122178731 IC50 > 30000 nM T96079 CU7TK1 122178732 IC50 > 30000 nM T96079 C5IC8D 122192916 IC50 = 255 nM T96079 CX4FJ9 122192917 IC50 = 1200 nM T96079 CZ19KN 122192918 IC50 = 130 nM T96079 CS5J0Y 122192922 IC50 = 35 nM T96079 C32JLB 122192923 IC50 = 18 nM T96079 CEJA32 122192964 IC50 = 2 nM T96079 C2M3HZ 122192965 IC50 = 23 nM T96079 C7PY6D 122192966 IC50 = 71 nM T96079 CFW2X9 122192967 IC50 = 39 nM T96079 CP80SV 122192968 IC50 = 2 nM T96079 CAC9G7 122192969 IC50 = 21000 nM T96079 CV1B7G 122193010 IC50 = 44 nM T96079 CJ6RO8 122193596 IC50 > 10000 nM T96079 CFX23Z 122193608 IC50 = 86 nM T96079 CF9OC5 127044948 IC50 = 1 nM T96079 C5JTD2 131801411 IC50 = 6 nM T96079 C26GLM 132578413 IC50 = 19.6 nM T96079 C2GK9S 132578414 IC50 = 35.7 nM T96079 CZC7S8 133081963 IC50 = 15.5 nM T96079 C7WUQ8 134132563 EC50 > 100000 nM T96079 CH0Z1F 134132933 IC50 = 18 nM T96079 CLJ42B 134133393 IC50 > 10000 nM T96079 C0KPZ2 134134008 EC50 = 56 nM T96079 CH8Y4O 134134119 EC50 = 62 nM T96079 CA82NT 134134445 EC50 < 100000 nM T96079 CL98GE 134134766 EC50 = 144 nM T96079 CWCT62 134135404 EC50 = 81 nM T96079 C4GH9N 134135423 EC50 = 52 nM T96079 CHCQ08 134135691 EC50 < 100000 nM T96079 CW57DV 134136045 IC50 > 10000 nM T96079 CZL9G5 134136499 IC50 = 282 nM T96079 CU21TD 134137235 IC50 = 222 nM T96079 CR2T3P 134137722 IC50 = 678 nM T96079 CSQA42 134137723 IC50 = 151 nM T96079 CTVU58 134137745 IC50 > 10000 nM T96079 C9TA4B 134138258 EC50 < 100000 nM T96079 C08GSU 134138415 EC50 < 100000 nM T96079 CJWI53 134138747 EC50 = 50 nM T96079 CG10OP 134138899 IC50 = 171 nM T96079 CMK0P1 134139045 EC50 > 100000 nM T96079 CX9T2Z 134139204 IC50 = 267 nM T96079 CB4SJ6 134139386 IC50 = 112 nM T96079 CZ8UX7 134139921 IC50 = 353 nM T96079 C56JXK 134140613 IC50 > 10000 nM T96079 CRP27O 134140664 EC50 = 92 nM T96079 CMV8X2 134140767 IC50 = 102 nM T96079 C3D2RJ 134141065 IC50 > 10000 nM T96079 C23TOG 134141938 EC50 > 100000 nM T96079 CV21FX 134142005 EC50 > 100000 nM T96079 C8H4NP 134142550 EC50 = 40 nM T96079 CT9U5R 134142869 IC50 = 1230 nM T96079 CVX04T 134143037 IC50 > 10000 nM T96079 C2Z3WL 134143183 EC50 = 111 nM T96079 CT7E6S 134143738 IC50 = 95 nM T96079 CX91FY 134144151 IC50 = 34 nM T96079 C58XGY 134144488 EC50 = 61000 nM T96079 C5NL0F 134144508 IC50 = 5900 nM T96079 CC5UV4 134145289 IC50 = 230 nM T96079 CGLT78 134145451 IC50 = 78 nM T96079 C0N2YL 134145647 IC50 > 10000 nM T96079 C4OK8J 134146914 EC50 = 83 nM T96079 CMAS93 134148082 IC50 > 10000 nM T96079 CS3AL8 134148939 EC50 > 100000 nM T96079 CWRA28 134150065 EC50 = 61 nM T96079 CB9EP8 134150735 IC50 = 137 nM T96079 CF6Z3S 134151621 EC50 = 65 nM T96079 CY25RS 134151866 IC50 > 10000 nM T96079 CLQN31 134152789 EC50 = 58 nM T96079 CTFG28 134153941 IC50 = 64 nM T96079 CR0MS7 134154190 IC50 = 73 nM T96079 CSU50Z 134154825 EC50 < 100000 nM T96079 CU3L7Q 134155140 EC50 = 74 nM T96079 CC01IU 134155143 IC50 = 548 nM T96079 CN26RH 134156666 IC50 = 127 nM T96079 CTO07X 134157327 IC50 = 5900 nM T96079 CZE6U4 134157900 IC50 = 131 nM T96079 CA8K9J 134157934 EC50 = 15 nM T96079 CWS04J 134158362 IC50 = 3200 nM T96079 CLD78B 134694953 Ki = 11000 nM T96079 CH9RX5 135313574 IC50 = 60.5 nM T96079 C2DP1L 135313576 IC50 = 62 nM T96079 CCJ97K 135313618 IC50 = 661 nM T96079 C76OJC 135313705 IC50 = 4316 nM T96079 C2L6PH 135313715 IC50 = 286 nM T96079 CO4W2L 135313730 IC50 = 25.2 nM T96079 CN7U0V 135313757 IC50 = 3307 nM T96079 C0G6IE 135313758 IC50 = 21 nM T96079 CD5FU8 135313764 IC50 = 1855 nM T96079 CQBZ60 135313773 IC50 = 292 nM T96079 C74VEJ 135313789 IC50 = 5751 nM T96079 CO7AJ2 135313829 IC50 = 8721 nM T96079 C3K2RL 135313899 IC50 = 143 nM T96079 C10GDT 135313911 IC50 = 698 nM T96079 CMR34P 135313919 IC50 = 45 nM T96079 CJAQ57 135313931 IC50 = 230 nM T96079 CQR2M1 135313955 IC50 = 163 nM T96079 CS5HY9 135313960 IC50 = 24 nM T96079 CR6K4Q 135313963 IC50 = 82.1 nM T96079 C9FNU5 135313965 IC50 = 1199 nM T96079 CQ4B1T 135313976 IC50 = 2902 nM T96079 CD8B0A 135313980 IC50 = 260 nM T96079 CGPC70 135313983 IC50 > 33000 nM T96079 C75MZN 135314048 IC50 = 16.1 nM T96079 CUA3M7 135314064 IC50 > 23000 nM T96079 CL12JU 135314107 IC50 = 91.2 nM T96079 CPTO20 135314108 IC50 = 21.4 nM T96079 C1XSQ4 135314132 IC50 = 1710 nM T96079 C8Q4JP 135314141 IC50 = 24.2 nM T96079 CFD5N1 135314164 IC50 > 33000 nM T96079 C63BWA 135314215 IC50 = 71 nM T96079 C57HTM 135314218 IC50 = 323 nM T96079 CXN1C7 135314251 IC50 = 58.3 nM T96079 CBQ01J 135314252 IC50 = 92.8 nM T96079 CU67EM 135314256 IC50 = 2116 nM T96079 CL23RS 135314305 IC50 = 69 nM T96079 CMC3E1 135314326 IC50 = 631 nM T96079 C9OZ3G 135314329 IC50 = 64.6 nM T96079 C46IBJ 135314337 IC50 = 90.3 nM T96079 CWI13E 135314362 IC50 = 510 nM T96079 CL6FK9 135314383 IC50 > 33000 nM T96079 CI73PJ 135314386 IC50 = 134 nM T96079 CM3KV6 135314388 IC50 = 115 nM T96079 CY24QI 135314390 IC50 = 40.7 nM T96079 CD64BJ 135314469 IC50 = 183 nM T96079 C3SM8K 137631624 IC50 > 30000 nM T96079 C02MSJ 137632194 IC50 > 30000 nM T96079 CC8N0O 137632426 IC50 = 210 nM T96079 CU1H0F 137632681 IC50 > 30000 nM T96079 CZJ72H 137632745 IC50 = 23.9 nM T96079 CJ2ZF8 137633110 IC50 = 72 nM T96079 C6MRU3 137633431 IC50 = 54.7 nM T96079 CV8M3P 137633531 IC50 = 36.3 nM T96079 CKI7E3 137634082 IC50 > 30000 nM T96079 CNU3O7 137634107 IC50 = 69.6 nM T96079 C1S2YN 137634372 IC50 > 30000 nM T96079 COD07I 137634464 IC50 = 77.6 nM T96079 CQS70B 137634879 IC50 > 30000 nM T96079 CT8E0M 137635041 IC50 = 3.71 nM T96079 CT8YI0 137635322 IC50 > 30000 nM T96079 C0V9CY 137636041 IC50 > 30000 nM T96079 CG84FX 137636198 IC50 > 30000 nM T96079 C8GLY9 137636313 IC50 > 30000 nM T96079 C51ALD 137636455 IC50 > 30000 nM T96079 CM9YP4 137636536 IC50 > 30000 nM T96079 C9YJ7H 137636951 IC50 = 6 nM T96079 CNM9G7 137637211 IC50 = 147.1 nM T96079 C8VM6G 137637238 IC50 = 25.6 nM T96079 CGB85J 137637266 IC50 = 22 nM T96079 CX91ZF 137637457 IC50 = 1530 nM T96079 C6A4JC 137637520 IC50 > 30000 nM T96079 C70RZU 137637646 IC50 = 180 nM T96079 C4T7AF 137637674 IC50 > 30000 nM T96079 CDBT63 137637838 IC50 = 20.1 nM T96079 CIZ7H9 137637865 IC50 > 10000 nM T96079 CLCG42 137638059 IC50 > 30000 nM T96079 C49CAF 137638093 IC50 > 30000 nM T96079 C21YPG 137638242 IC50 = 15.3 nM T96079 CQ9PI1 137638674 IC50 > 30000 nM T96079 CI7Z8T 137638711 IC50 = 859.7 nM T96079 CH64ZI 137638861 IC50 = 2140 nM T96079 CF8S5N 137639002 Ki > 6200 nM T96079 CTV94W 137639137 IC50 > 30000 nM T96079 C8WO2G 137639251 IC50 = 17 nM T96079 CMF9Q1 137639293 IC50 > 30000 nM T96079 C6D1AF 137639743 IC50 > 30000 nM T96079 C9V0MW 137639865 IC50 > 10000 nM T96079 CYPQ38 137640446 IC50 = 43.8 nM T96079 C2J8YF 137640469 IC50 = 3690 nM T96079 CV85YQ 137640474 IC50 = 52.9 nM T96079 C1OG4M 137640505 IC50 > 30000 nM T96079 CB5L0M 137640842 IC50 = 21000 nM T96079 C0Q4IM 137641652 IC50 = 63.4 nM T96079 CYW61U 137641749 IC50 = 129 nM T96079 C19LKY 137642595 IC50 = 46.8 nM T96079 CM8TG3 137643051 IC50 = 72.2 nM T96079 CWEM42 137643115 IC50 = 70.4 nM T96079 CVC3S2 137643317 IC50 = 29.4 nM T96079 CO01IW 137643816 IC50 > 30000 nM T96079 C4S3JQ 137643895 IC50 > 10000 nM T96079 C31KCL 137644260 IC50 > 30000 nM T96079 CI2F1B 137644335 IC50 = 664 nM T96079 CW7R9J 137644796 IC50 > 30000 nM T96079 CU91LQ 137644813 IC50 = 541 nM T96079 CYI0F2 137644874 IC50 > 30000 nM T96079 CB78AN 137644938 IC50 > 30000 nM T96079 C78HFG 137645641 IC50 > 30000 nM T96079 C8DF4P 137645906 IC50 > 30000 nM T96079 CKT2R4 137646125 IC50 = 158 nM T96079 CL8AG9 137646518 IC50 = 472.7 nM T96079 CF14IB 137646840 IC50 > 30000 nM T96079 CRA48Q 137647184 EC50 > 30000 nM T96079 CXS2U7 137647336 IC50 = 50.8 nM T96079 CT8HC6 137647496 IC50 > 10000 nM T96079 C42DRJ 137647643 IC50 = 471 nM T96079 CLAR76 137647645 IC50 = 45.5 nM T96079 C4AKD7 137647838 IC50 = 24.6 nM T96079 CT86OF 137647937 IC50 > 30000 nM T96079 CA42ZD 137648113 IC50 = 91.6 nM T96079 C5ZP8U 137648152 IC50 > 30000 nM T96079 C4DY6Z 137648169 IC50 > 30000 nM T96079 CJW62B 137648362 IC50 = 81.8 nM T96079 CPJV29 137648481 IC50 > 30000 nM T96079 CM56QZ 137648951 IC50 = 1.5 nM T96079 CCT4L9 137649106 IC50 > 30000 nM T96079 CBFO36 137649245 IC50 = 61.1 nM T96079 CE84CA 137649371 IC50 = 47.8 nM T96079 CZ4S8Y 137649869 IC50 = 88.5 nM T96079 CH7MV8 137650158 IC50 > 30000 nM T96079 CRP80C 137650276 IC50 > 30000 nM T96079 C28PSD 137651290 IC50 = 1250 nM T96079 CD9ZN4 137651429 IC50 = 36.5 nM T96079 CC75QA 137651588 IC50 > 30000 nM T96079 C1RN3A 137651859 IC50 = 360 nM T96079 CRH02L 137652168 IC50 > 30000 nM T96079 C2L7ZT 137652982 IC50 = 22.7 nM T96079 CNOX24 137653243 IC50 > 30000 nM T96079 CJFE85 137653778 IC50 > 10000 nM T96079 CY2L4S 137653914 IC50 > 10000 nM T96079 C4L1JP 137654103 IC50 = 1800 nM T96079 CV59RY 137654290 IC50 = 168 nM T96079 CQL18X 137654477 IC50 = 70 nM T96079 CV35EJ 137654804 IC50 > 30000 nM T96079 CE6L3M 137655149 IC50 > 30000 nM T96079 CUC1D4 137655552 IC50 > 30000 nM T96079 C65MBR 137655630 IC50 = 17000 nM T96079 C5S3IL 137655887 IC50 > 30000 nM T96079 C25RWZ 137655917 IC50 > 30000 nM T96079 CRY40J 137655938 IC50 = 9.26 nM T96079 CNU89M 137656325 IC50 > 30000 nM T96079 C29UVL 137656780 EC50 > 30000 nM T96079 CN4C2T 137657155 IC50 > 30000 nM T96079 C8DT1W 137657247 IC50 = 69 nM T96079 CUQ12W 137657505 IC50 > 10000 nM T96079 C2BGF3 137657547 IC50 = 832 nM T96079 CZ70YL 137658374 IC50 > 30000 nM T96079 C35DVM 137658485 IC50 = 72.1 nM T96079 CHZ2Y8 137658540 IC50 = 82.6 nM T96079 C1R7UP 137658901 IC50 = 168 nM T96079 C1VZ2U 137659906 IC50 > 30000 nM T96079 CH9A8Q 137660298 IC50 = 10000 nM T96079 C1R5BU 137660760 IC50 > 30000 nM T96079 C51FPJ 137660789 IC50 > 30000 nM T96079 C9M7JB 137660814 IC50 > 30000 nM T96079 C1K4GE 137660848 IC50 = 399.3 nM T96079 CAP85L 137660893 IC50 > 30000 nM T96079 CXK05E 137661256 IC50 > 10000 nM T96079 CT6KM9 137661467 IC50 > 30000 nM T96079 CSEZ59 137662026 IC50 = 75.2 nM T96079 C5Q8UM 137662063 IC50 > 30000 nM T96079 C2HLM9 137662117 IC50 = 708.3 nM T96079 C2VRA9 137662172 IC50 > 30000 nM T96079 C3W2AE 138491830 IC50 = 180 nM T96079 CA8H1N 138491848 IC50 > 10000 nM T96079 CD74JM 138491853 IC50 > 10000 nM T96079 C7E3LH 138501771 IC50 > 10000 nM T96079 CAF0S2 138501773 IC50 > 10000 nM T96079 C29VUI 138501774 IC50 > 10000 nM T96079 CYDF05 142416702 IC50 = 127 nM T96079 C06ZBJ 142416740 IC50 = 171 nM T96079 C9J1ZO 142416754 IC50 = 98 nM T96079 CZA08U 142416759 IC50 = 406 nM T96079 C58KQF 142416884 IC50 = 34 nM T96079 C68OXK 142416914 IC50 = 1800 nM T96079 C7C3MK 142416935 IC50 = 381 nM T96079 CO7DK2 142416967 IC50 = 280 nM T96079 CVND41 145949156 IC50 = 1154 nM T96079 CI14LP 145949343 IC50 = 16 nM T96079 C8KA6P 145949486 IC50 = 17 nM T96079 CA0B3D 145949907 IC50 = 195 nM T96079 C7W9ZT 145949949 IC50 = 364 nM T96079 CAT5E1 145950272 IC50 = 6 nM T96079 COG04E 145950432 IC50 = 80 nM T96079 CAWU95 145950510 IC50 = 16.9 nM T96079 CL2OR1 145950976 IC50 = 6.08 nM T96079 C2M8PI 145951236 IC50 = 2.92 nM T96079 CJ9OT7 145951410 IC50 = 190 nM T96079 C3OMF2 145951963 IC50 = 44 nM T96079 CC4K9F 145952601 IC50 = 171 nM T96079 CGW92C 145952721 IC50 = 17 nM T96079 C2FXL5 145952723 IC50 = 30.7 nM T96079 CER83S 145953040 IC50 = 14.8 nM T96079 C1A4CH 145953177 IC50 = 23.5 nM T96079 COZ1F4 145953325 IC50 = 32 nM T96079 C09WNF 145953342 IC50 = 553 nM T96079 CEJ26X 145953403 IC50 = 50 nM T96079 CS21ZB 145953739 IC50 = 536 nM T96079 CXQ8V3 145953887 IC50 = 120 nM T96079 CPW52X 145954567 IC50 = 230 nM T96079 C59AVT 145954818 IC50 = 29.6 nM T96079 C4P6MT 145954878 IC50 = 17.9 nM T96079 CK0S1G 145955694 IC50 = 2639 nM T96079 CE03RK 145955745 IC50 = 498 nM T96079 CF6T7G 145955884 IC50 = 26.7 nM T96079 C0HN4S 145955917 IC50 = 340 nM T96079 C8Y4VT 145956312 IC50 = 14.1 nM T96079 CXAR52 145956817 IC50 = 11 nM T96079 C4G6XJ 145956824 IC50 = 13 nM T96079 CQ0JP4 145957239 IC50 = 313 nM T96079 CK94HO 145957365 IC50 = 65 nM T96079 C70LMY 145957553 IC50 = 13.8 nM T96079 CB2K0W 145957599 IC50 = 4.47 nM T96079 C2YIB0 145958083 EC50 = 9549.93 nM T96079 C8WZY3 145958093 IC50 = 66 nM T96079 CXHM49 145958111 IC50 = 8.6 nM T96079 CO4EU0 145958234 IC50 = 11 nM T96079 CBC1T9 145958296 IC50 = 28 nM T96079 C3TX8O 145958528 IC50 = 161 nM T96079 CT3U1A 145958698 EC50 > 30000 nM T96079 CH47WN 145959135 IC50 = 210 nM T96079 CW8M0I 145959142 IC50 = 61 nM T96079 C8DH5F 145959814 IC50 = 150 nM T96079 C5Z9US 145959844 IC50 = 125 nM T96079 CUD9E6 145960079 IC50 = 33.9 nM T96079 CI8Q2V 145960175 IC50 = 28 nM T96079 C3F8XM 145960247 IC50 = 20.7 nM T96079 C6C5JX 145961199 IC50 = 1000 nM T96079 CD01PX 145961863 IC50 = 959 nM T96079 C64OLM 145963140 IC50 = 3.59 nM T96079 CU8Y2C 145963537 IC50 = 62 nM T96079 C57KNJ 145964516 IC50 = 2600 nM T96079 CWJE58 145965128 IC50 = 1020 nM T96079 C9VG0C 145965140 IC50 > 10000 nM T96079 CX0BZ7 145966697 IC50 = 170 nM T96079 CBZ29Q 145969178 IC50 = 640 nM T96079 CND2K7 145971189 IC50 = 33 nM T96079 CMI45E 145971507 IC50 = 32.2 nM T96079 CK56QO 145972040 IC50 = 18 nM T96079 C7UJS2 145972313 IC50 = 68 nM T96079 C2G0VR 145972431 EC50 = 5888.44 nM T96079 CL72KB 145972839 IC50 = 210 nM T96079 CP7LW2 145973146 IC50 = 715 nM T96079 C8OSM0 145973345 IC50 = 146 nM T96079 CRYM18 145973908 IC50 = 54 nM T96079 C54QHK 145974080 IC50 = 154 nM T96079 C09EUQ 145974150 IC50 = 1050 nM T96079 C94RWZ 145974553 IC50 = 190 nM T96079 CP20BX 145974804 IC50 = 484 nM T96079 CBEJ75 145975500 IC50 = 630 nM T96079 CF91PL 145975537 IC50 = 18 nM T96079 CH30YP 145975799 IC50 = 88 nM T96079 CB1X0G 145975925 IC50 = 290 nM T96079 CEU3V9 145976370 IC50 < 20 nM T96079 CMYH51 145976437 IC50 = 200 nM T96079 CCR1F0 145976496 IC50 = 320 nM T96079 C2HTM6 145977928 IC50 = 150 nM T96079 CE0K5V 155511299 IC50 = 747 nM T96079 C8Z1JT 155513322 IC50 = 501.19 nM T96079 C4EBX9 155513527 IC50 = 501.19 nM T96079 C1RO9S 155513627 IC50 = 1560 nM T96079 CI4DQ0 155514823 IC50 = 794.33 nM T96079 CAS9E6 155515208 IC50 = 193 nM T96079 C5AX9S 155516007 IC50 > 10000 nM T96079 C5C8DT 155516872 IC50 = 22 nM T96079 C6ZK8M 155517509 IC50 = 7418 nM T96079 CG4WK9 155517575 IC50 = 251.19 nM T96079 C2ELM4 155518071 IC50 = 630.96 nM T96079 C2JKU5 155518667 IC50 = 2000 nM T96079 CC3H4U 155518713 IC50 = 9700 nM T96079 C4H2DQ 155519352 IC50 > 10000 nM T96079 C2LS4J 155519637 IC50 > 10000 nM T96079 CR35QE 155519969 IC50 = 2900 nM T96079 CXN46O 155521148 IC50 = 2511.89 nM T96079 CJHC74 155521886 IC50 = 407 nM T96079 CC60BA 155521909 IC50 = 3.5 nM T96079 CZT8X5 155522667 IC50 > 50000 nM T96079 CCH9O2 155523400 IC50 = 158.49 nM T96079 C49HKA 155525671 IC50 = 1.6 nM T96079 C4YWV9 155525712 IC50 = 9900 nM T96079 C3HGV5 155526368 IC50 > 10000 nM T96079 CN13EB 155527692 IC50 = 10000 nM T96079 C7F8DY 155528475 IC50 = 2200 nM T96079 CQ7JD5 155529936 IC50 = 251.19 nM T96079 C4GI2E 155529939 IC50 = 1258.93 nM T96079 C3BV0S 155530073 IC50 = 8800 nM T96079 CNZ0M4 155530935 IC50 = 2511.89 nM T96079 CHE2I9 155531953 IC50 = 8700 nM T96079 CUM2C7 155534351 IC50 = 737 nM T96079 CVU9O6 155534395 IC50 = 147 nM T96079 CNW62I 155534587 IC50 = 23 nM T96079 CX4Q7O 155534825 IC50 = 64 nM T96079 C0C2YJ 155534891 IC50 > 1000 nM T96079 C8HM6F 155535518 IC50 = 8800 nM T96079 CDB2A4 155535988 IC50 > 10000 nM T96079 C05UQJ 155537257 IC50 = 8600 nM T96079 COFA71 155537468 IC50 = 25 nM T96079 C16VIH 155537796 IC50 > 1000 nM T96079 CW1F7Y 155538284 IC50 = 5600 nM T96079 C43DZF 155538662 IC50 > 10000 nM T96079 CA5W8S 155539331 IC50 = 316.23 nM T96079 CAR9V8 155542313 IC50 = 502 nM T96079 CG1A6D 155542701 IC50 = 18 nM T96079 C8OUE7 155543253 IC50 > 1000 nM T96079 CG6VC8 155543662 IC50 > 10000 nM T96079 CYMI50 155544179 IC50 = 1995.26 nM T96079 CFR62J 155544237 IC50 > 10000 nM T96079 CAL93B 155544593 IC50 = 615 nM T96079 C5RY1V 155545540 IC50 = 1000 nM T96079 CH17YG 155545664 IC50 = 4.5 nM T96079 CGOA27 155546069 IC50 > 10000 nM T96079 C1JUO3 155546536 IC50 = 32 nM T96079 C29EWJ 155546592 IC50 = 10 nM T96079 C2PE7M 155546659 IC50 > 10000 nM T96079 C07KFL 155547373 IC50 = 199.53 nM T96079 CV3C0R 155548895 IC50 = 5.7 nM T96079 C3M2QO 155548932 IC50 > 10000 nM T96079 CC5P4D 155549012 IC50 = 794.33 nM T96079 C0XEJ7 155550204 IC50 > 10000 nM T96079 C1SG8P 155550210 IC50 = 794.33 nM T96079 CW4D3J 155550367 IC50 = 5500 nM T96079 C9LM2O 155551009 IC50 > 1000 nM T96079 C0W6YM 155551439 IC50 = 14 nM T96079 C04LBX 155554725 IC50 = 316.23 nM T96079 CU5XR3 155554813 IC50 = 9600 nM T96079 C2THI9 155554828 IC50 > 10000 nM T96079 CHXL93 155554948 IC50 = 462 nM T96079 CW8H5K 155556244 IC50 > 1000 nM T96079 CXK6O9 155557524 IC50 = 251.19 nM T96079 CDT78C 155558601 IC50 > 3000 nM T96079 C5S8PU 155558653 IC50 = 34 nM T96079 CUDX85 155558835 IC50 = 1000 nM T96079 CDN52W 155559655 IC50 > 1000 nM T96079 CYEO80 155560189 IC50 = 474 nM T96079 CUPI87 155560382 IC50 = 7.9 nM T96079 CS4C9P 155560529 IC50 = 110 nM T96079 CN3U1L 155561023 IC50 > 10000 nM T96079 C1C7HN 155561098 IC50 = 3162.28 nM T96079 CB0QO6 155562280 IC50 = 2511.89 nM T96079 C8X6CV 155562705 IC50 > 1000 nM T96079 C0YOS1 155563693 IC50 > 10000 nM T96079 C3EKH7 155564611 IC50 > 10000 nM T96079 CK1FC9 155566596 IC50 = 144 nM T96079 CM57PG 155566843 IC50 = 316.23 nM T96079 C6OES3 155567133 IC50 = 3900 nM T96079 CU2PA1 155568737 IC50 > 1000 nM T96079 CMG5R7 155569501 IC50 = 3500 nM T96079 D00GII 44418888 IC50 = 99 nM T96079 D00XBM 44418891 IC50 = 157 nM T96079 D02UES 44418892 IC50 = 3 nM T96079 D03QJA 11718722 IC50 = 0.87 nM T96079 D04BVW 44418894 IC50 = 563 nM T96079 D04PDF 44418872 IC50 = 170 nM T96079 D04TED 44418887 IC50 = 23 nM T96079 D04TIO 5275843 IC50 = 4 nM T96079 D04XHX 44418885 IC50 = 350 nM T96079 D05VQJ 25147749 IC50 = 8 nM T96079 D05YHT 44418895 IC50 = 256 nM T96079 D06MBD 11176403 IC50 = 11 nM T96079 D08XRM 44418890 IC50 = 167 nM T96079 D08YYV 44418893 IC50 = 21 nM T96079 D0B8VW 44418889 IC50 = 250 nM T96079 D0BH8K 44418879 IC50 = 92 nM T96079 D0FQ3G 44418869 IC50 = 230 nM T96079 D0K0SO 44418880 IC50 = 11 nM T96079 D0K9KQ 44418868 IC50 = 130 nM T96079 D0M6RQ 44418865 IC50 = 63 nM T96079 D0P7UV 44418878 IC50 = 47 nM T96079 D0Q3MM 11158428 IC50 = 4 nM T96079 D0S0GV 44418886 IC50 = 128 nM T96079 D0S0PU 44418873 IC50 = 11 nM T96079 D0ST1U 44418883 IC50 = 640 nM T96079 D0ZO3C 11331592 IC50 = 8 nM T88699 CSNX56 496 Ki = 1370000 nM T88699 COJ39Y 4026 Ki = 90 nM T88699 C6K1JO 122356 Ki = 800000 nM T88699 CZ3H8A 129689 Ki = 180 nM T88699 CCBA97 146442 Ki = 300 nM T88699 CYK6W9 162081 Ki = 31000 nM T88699 CMLD96 4194799 Ki = 110000 nM T88699 C1D9PK 4420356 Ki = 75000 nM T88699 CG7AB9 13561211 Ki = 700 nM T88699 CW4BV9 14484861 Ki = 29000000 nM T88699 CHAQ24 14484863 Ki = 26000 nM T88699 CKF4I6 14484867 Ki = 376000 nM T88699 C35KED 14484869 Ki = 650000 nM T88699 C6EJQ5 14484872 Ki = 260000 nM T88699 C5QHE6 14484874 Ki = 130000 nM T88699 C50DXA 14484877 Ki = 96 nM T88699 C4V1AQ 14484879 Ki = 100 nM T88699 CI89TC 14484881 Ki = 630 nM T88699 CN7JT4 14484883 Ki = 1000 nM T88699 C62LXZ 17772784 Ki = 2200 nM T88699 CU0W6Z 44302492 Ki = 425000 nM T88699 C4WKF3 44302512 Ki = 310000 nM T88699 CM7R6T 123440770 IC50 > 200000 nM T88699 C2BGD3 155513276 IC50 > 200000 nM T88699 CUI18M 155515157 IC50 > 200000 nM T88699 CPU41A 155528785 IC50 > 200000 nM T88699 CV5TY2 155535062 IC50 > 200000 nM T88699 CB6W7X 155538837 IC50 > 200000 nM T88699 CPXY64 155544313 IC50 > 200000 nM T88699 CEF57Y 155551313 IC50 > 200000 nM T88699 CF1CQ9 155553798 IC50 > 200000 nM T88699 C2BH3L 155561208 IC50 > 200000 nM T88699 C9Q7WZ 155567401 IC50 > 200000 nM T31595 D00NPP 60855 IC50 = 0.8 nM T31595 D0C4YC 4075 IC50 > 100000 nM T31595 D0P2IW 154234 IC50 = 0.4 nM T31595 C3RJ7D 6844 IC50 > 100000 nM T31595 C9JK2Q 490476 IC50 = 1 nM T31595 CN26ID 643181 IC50 > 100000 nM T31595 CY7C5W 23626540 IC50 = 0.09 nM T31595 CJ63EC 25225410 IC50 > 3000 nM T31595 CU45XW 25225411 IC50 = 1679 nM T31595 CJEQ27 25225622 IC50 = 1.1 nM T31595 CJ1PY3 44123802 IC50 = 1719 nM T31595 CO1K3W 53484070 IC50 = 590 nM T31595 CM95RC 58753598 IC50 = 0.99 nM T31595 CL3DZ8 71450551 IC50 = 2.9 nM T31595 CH0MK4 71450552 IC50 = 11.7 nM T31595 CZO89L 71454165 IC50 = 41.3 nM T31595 C73CRB 71454203 IC50 = 996 nM T31595 C4BUR6 71455897 IC50 = 3986 nM T31595 CUT28E 71457693 IC50 = 8.6 nM T31595 CB0GP3 71457694 IC50 = 3.1 nM T31595 CT3V1Z 71459606 IC50 = 2.9 nM T31595 C24ZDL 71461345 IC50 = 5.4 nM T31595 C42LDJ 71461346 IC50 = 0.7 nM T31595 C1LH0E 71463064 IC50 = 2853 nM T31595 C6ZAD2 71723924 IC50 = 20 nM T31595 C10FJD 71811523 IC50 = 200 nM T31595 C7X4HB 71811563 IC50 = 0.9 nM T31595 CE3M9C 90643657 IC50 = 1443 nM T31595 CW57MV 90643658 IC50 = 1283 nM T31595 CKB82W 90643660 IC50 = 10.9 nM T31595 CVN90R 90643661 IC50 = 89.2 nM T31595 CKBY53 90643662 IC50 = 24.6 nM T31595 CIP04R 118722031 IC50 = 6648 nM T31595 CTDY57 118722032 IC50 = 1010 nM T31595 CJW5Z2 118722033 IC50 = 1108 nM T31595 CX76VT 118722034 IC50 = 781 nM T31595 CW37HJ 118722035 IC50 = 6946 nM T31595 CY9OX2 118722036 IC50 = 1227 nM T31595 C3QD2F 118722037 IC50 = 19085 nM T31595 CY9CV1 118722041 IC50 = 19.5 nM T31595 C2YDR4 118722042 IC50 = 832 nM T31595 CF1VG7 118722043 IC50 = 1108 nM T31595 CYW6A4 118722044 IC50 = 13399 nM T31595 CLHW01 134135159 IC50 = 146.2 nM T31595 C7WYM1 134137939 IC50 = 238.3 nM T31595 CT3FK6 134138789 IC50 = 8 nM T31595 CX1W6P 134140037 IC50 = 31 nM T31595 CMWV70 134141175 IC50 = 9.9 nM T31595 CZ9U1B 134141213 IC50 = 12 nM T31595 CV9R2O 134141975 IC50 = 15 nM T31595 C4VJ5M 134142942 IC50 = 168.6 nM T31595 C59KYU 134143842 IC50 = 14 nM T31595 C26HRN 134144448 IC50 = 14 nM T31595 C5YO3J 134144783 IC50 = 15 nM T31595 CJ40KR 134146669 IC50 = 13 nM T31595 C8U1ZF 134146944 IC50 = 29 nM T31595 CE3Y4Q 134148983 IC50 = 12 nM T31595 CY9D1B 134150391 IC50 = 12 nM T31595 CSI6K3 134153666 IC50 = 2.3 nM T31595 CNS2O1 134153678 IC50 = 10 nM T31595 C4YN0Q 134157256 IC50 = 9 nM T31595 COS71V 145950310 IC50 = 8 nM T31595 CGL49X 145956701 IC50 = 53 nM T31595 CC7F3B 145959178 IC50 = 180 nM T31595 C0Q9NK 145973579 IC50 > 100000 nM T31595 CK7B1X 145980919 IC50 = 0.67 nM T31595 C1BJH2 145988356 IC50 = 0.94 nM T31595 CQ45WF 145989983 IC50 = 0.64 nM T31595 CN9QL7 145990747 IC50 = 0.44 nM T31595 D06IDO 449381 IC50 = 2.6 nM T31595 D0V9EN 689043 IC50 > 100000 nM T31595 D0YN3T 10336127 IC50 = 2.4 nM T31946 D07POC 176870 IC50 = 250 nM T31946 D0G6QF 3081361 IC50 = 25 nM T31946 D03AND 11656518 IC50 = 20 nM T31946 D0P6DJ 151194 IC50 = 100 nM T31946 D0VF6E 1401 IC50 = 190 nM T31946 D0L5YF 5329032 IC50 = 50 nM T31946 C8W3LH 286220 IC50 = 22000 nM T31946 CPN2S0 4369497 IC50 = 370 nM T31946 CB3G6R 4913175 IC50 = 100 nM T31946 CWX63A 5329004 IC50 = 37 nM T31946 CZU0K3 5329011 IC50 = 40 nM T31946 CJ68OQ 5329013 IC50 = 4 nM T31946 C1XJL0 5329019 IC50 = 300 nM T31946 C9SZ4Q 5329020 IC50 = 50 nM T31946 C3VHF6 5329026 IC50 = 200 nM T31946 CB6V5Y 5329028 IC50 = 40 nM T31946 C4VLR8 5329033 IC50 = 20 nM T31946 CLT7J9 5329034 IC50 = 600 nM T31946 C9VX8C 5329040 IC50 = 500 nM T31946 CK6T4U 5329042 IC50 = 65 nM T31946 CA81XO 5329045 IC50 = 60 nM T31946 C4T3MO 5329046 IC50 = 100 nM T31946 CQ15KR 5329049 IC50 = 250 nM T31946 C49KNS 5329050 IC50 = 100 nM T31946 C3C1EZ 5329051 IC50 = 70 nM T31946 C0H5XL 5329052 IC50 = 70 nM T31946 CW0KA8 5329053 IC50 = 60 nM T31946 COEN93 5329054 IC50 = 40 nM T31946 CATX52 5329055 IC50 = 80 nM T31946 CEQP41 5329056 IC50 = 60 nM T31946 CDV4C9 5329057 IC50 = 40 nM T31946 CNYT34 5329364 IC50 = 1410 nM T31946 C9ZPN1 5329365 IC50 = 495 nM T31946 CFDU12 5329366 IC50 = 328 nM T31946 CH19WM 5329368 IC50 = 256 nM T31946 CYN3I2 5329415 IC50 = 151 nM T31946 COM81Z 5329417 IC50 = 19 nM T31946 CKF1O7 5329419 IC50 = 88 nM T31946 C7WEG5 5329421 IC50 = 22 nM T31946 CZP9C6 5329424 IC50 = 303 nM T31946 C9MZ2K 5329426 IC50 = 26 nM T31946 CU5IV8 5329428 IC50 = 23 nM T31946 CB8O7C 5329429 IC50 = 396 nM T31946 CI4TV0 5329446 IC50 = 22 nM T31946 CWYP60 5329447 IC50 = 32 nM T31946 C21ZFW 5329449 IC50 = 23 nM T31946 CKT02A 5329452 IC50 = 29 nM T31946 C4RUV5 5329453 IC50 = 31 nM T31946 CGN7B0 5329457 IC50 = 150 nM T31946 CFS3A4 5329467 IC50 = 127 nM T31946 CKR04W 5329469 IC50 = 70 nM T31946 C9Q1US 5329470 IC50 = 80 nM T31946 CRGY13 5329471 IC50 = 20 nM T31946 CL71UW 5329848 IC50 = 10200 nM T31946 CTI5D4 5329853 IC50 = 1690 nM T31946 CT3F6Z 5329854 IC50 = 420 nM T31946 CHL9K2 5329855 IC50 = 1310 nM T31946 CNX7V5 5329856 IC50 = 290 nM T31946 CB7Z8S 5329857 IC50 = 7600 nM T31946 C1TL9F 5329858 IC50 = 650 nM T31946 CKG85D 5329859 IC50 = 1620 nM T31946 CWQ0O8 5329860 IC50 = 1650 nM T31946 CF4X1J 5329861 IC50 = 350 nM T31946 C8TAE1 5329862 IC50 = 3200 nM T31946 C6KDO7 5329863 IC50 = 930 nM T31946 CL46MG 5329864 IC50 = 300 nM T31946 C9T3UE 5329865 IC50 = 490 nM T31946 CYS31K 5329866 IC50 = 210 nM T31946 CQ3B5A 5329867 IC50 = 1940 nM T31946 C38MLW 5329868 IC50 = 13900 nM T31946 C0ZG9W 5329869 IC50 = 260 nM T31946 CS1VJ5 5329870 IC50 = 140 nM T31946 CCL8O5 5329871 IC50 = 960 nM T31946 CQ8ZH5 5329872 IC50 = 15000 nM T31946 C32HVT 5329873 IC50 = 170 nM T31946 C7AZY0 5329874 IC50 = 110 nM T31946 C49TVA 5329875 IC50 = 40 nM T31946 CD0IV1 5329876 IC50 = 50 nM T31946 CNWK81 5330126 IC50 = 880 nM T31946 CV7GX5 5330127 IC50 = 73 nM T31946 CWAR90 5330128 IC50 = 280 nM T31946 CDG3Z1 5330129 IC50 = 82 nM T31946 C09VSN 5330130 IC50 = 66 nM T31946 CV4U8Y 5330132 IC50 = 530 nM T31946 C6D7WJ 5330133 IC50 = 43 nM T31946 C2UX4V 5330134 IC50 = 91 nM T31946 CWQ47D 5330136 IC50 = 190 nM T31946 CLI47K 5330157 IC50 = 47 nM T31946 CNI15R 5330158 IC50 = 41 nM T31946 C4IA7N 5330159 IC50 = 47 nM T31946 CW8G9J 5330166 IC50 = 930 nM T31946 C7Z2YH 5330167 IC50 = 220 nM T31946 CEX9A7 5330168 IC50 = 1800 nM T31946 C3I6KF 5330169 IC50 = 3000 nM T31946 CZ3LK2 5330387 IC50 = 5 nM T31946 C4A8RX 9794758 IC50 = 360000 nM T31946 C43FVO 9859850 IC50 = 98000 nM T31946 CM5Z8X 9869943 IC50 > 100000 nM T31946 CXA5C8 9893493 IC50 = 100 nM T31946 CHB0D2 9982235 IC50 = 6.7 nM T31946 CY04DA 10021712 IC50 = 170 nM T31946 C1JUF8 10073832 IC50 = 17 nM T31946 CCY2X5 10113563 IC50 = 200 nM T31946 CA31MX 10131256 IC50 = 213000 nM T31946 C1TX8D 10198953 IC50 = 477000 nM T31946 C2RLF5 10199254 IC50 = 310000 nM T31946 C7OA9P 10325135 IC50 = 62 nM T31946 C07XHY 10388612 IC50 = 1.1 nM T31946 C2VPT6 10436729 IC50 = 2.1 nM T31946 C7PLI5 10478569 IC50 = 7.6 nM T31946 COMB49 11155938 IC50 = 4 nM T31946 C7MOP5 11163572 IC50 = 16000 nM T31946 CG13KT 11164265 IC50 = 350 nM T31946 C0IZ1Q 11164266 IC50 = 910 nM T31946 CJ4F6C 11176518 IC50 = 410 nM T31946 C0U4FC 11181380 IC50 = 13000 nM T31946 CGEM63 11181426 IC50 = 1300 nM T31946 CXO79R 11181788 IC50 = 250 nM T31946 C1ID9O 11187999 IC50 = 5900 nM T31946 CJ17RV 11188442 IC50 = 3900 nM T31946 CC0IL6 11188738 IC50 = 460 nM T31946 C9BDW0 11188739 IC50 = 1400 nM T31946 C2FNC3 11193260 IC50 = 610 nM T31946 C0ER9P 11200665 IC50 = 250 nM T31946 CZ2XI3 11210965 IC50 = 560 nM T31946 CV52AN 11211004 IC50 = 930 nM T31946 C6Z4TS 11211061 IC50 = 910 nM T31946 CC97TS 11211990 IC50 = 11000 nM T31946 CE6T8H 11231939 IC50 = 3260 nM T31946 CKT2C3 11239220 IC50 = 2000 nM T31946 CB2XI8 11239299 IC50 = 620 nM T31946 CICX97 11244488 IC50 = 1130 nM T31946 C0A4EL 11244838 IC50 = 210 nM T31946 CX7K9G 11245472 IC50 = 440 nM T31946 C9K3HO 11245920 IC50 = 360 nM T31946 CLK02N 11248789 IC50 = 910 nM T31946 CM10OX 11262303 IC50 = 630 nM T31946 C1J9GW 11279720 IC50 > 20000 nM T31946 C8FGR1 11288910 IC50 > 2500000 nM T31946 C3Y0AT 11293142 IC50 > 20000 nM T31946 CP34IZ 11303701 IC50 = 13000 nM T31946 CE16IZ 11308204 IC50 = 3200 nM T31946 C37JZP 11314529 IC50 = 14000 nM T31946 CGMD57 11316827 IC50 = 31 nM T31946 C3YA8L 11318315 IC50 = 19 nM T31946 CC8J3N 11328182 IC50 = 50 nM T31946 CQF1S6 11331282 IC50 = 18000 nM T31946 CR3EN9 11331584 IC50 = 1400 nM T31946 CA6F4L 11352215 IC50 = 2.1 nM T31946 CDZR14 11357877 IC50 > 2500000 nM T31946 CYP41W 11371392 IC50 > 15000 nM T31946 CG57WD 11374515 IC50 = 1.8 nM T31946 C4H0ZP 11380375 IC50 > 2500000 nM T31946 CM30TC 11387552 IC50 < 10 nM T31946 C05CWH 11392350 IC50 = 7600 nM T31946 C8XWO5 11393780 IC50 = 750 nM T31946 CSG8Q4 11395135 IC50 = 16000 nM T31946 CT3BL8 11411362 IC50 = 4600 nM T31946 CQD35C 11419379 IC50 = 6.8 nM T31946 C7AI2V 11432911 IC50 = 27 nM T31946 CQB38J 11433537 IC50 = 2700 nM T31946 C6CN5S 11439660 IC50 = 10000 nM T31946 C7C8OJ 11441201 IC50 = 240 nM T31946 C45WKC 11442803 IC50 = 18 nM T31946 CG1UZ2 11445097 IC50 = 300 nM T31946 C9SO0A 11451977 IC50 = 350 nM T31946 CZ9O1A 11455031 IC50 = 25 nM T31946 CM40XT 11462674 IC50 = 5900 nM T31946 CCZB40 11462990 IC50 = 1300 nM T31946 C8MY1P 11463998 IC50 > 20000 nM T31946 CJUF06 11464544 IC50 = 91 nM T31946 CTG3D9 11465545 IC50 = 3.6 nM T31946 C4V3NJ 11473497 IC50 = 410 nM T31946 CU4Z7Q 11474329 IC50 = 530 nM T31946 C3AG9S 11474703 IC50 = 1200 nM T31946 C6M9NC 11477626 IC50 = 46 nM T31946 C29DYA 11486622 IC50 > 20000 nM T31946 CE39WZ 11488852 IC50 = 35 nM T31946 CZI6D9 11493632 IC50 = 200 nM T31946 CD8G0U 11506240 IC50 = 40300 nM T31946 CGN83M 11544306 IC50 = 631 nM T31946 CE6P8L 11595868 IC50 = 3980 nM T31946 C65ZXO 11632139 IC50 = 251 nM T31946 CE5MY2 11645981 IC50 > 10000 nM T31946 C0UGQ3 11689490 IC50 = 3980 nM T31946 C1H6FA 11750102 IC50 = 970 nM T31946 CFY5A0 11750103 IC50 = 1400 nM T31946 C2EPQ0 11763954 IC50 = 240 nM T31946 CTP2M1 11772795 IC50 = 9900 nM T31946 C4Q1AE 11817879 IC50 > 2500000 nM T31946 CFKE48 16064750 IC50 = 70 nM T31946 CFN6G4 21701597 IC50 = 50 nM T31946 CGX61W 22041319 IC50 = 5 nM T31946 CF6LA9 22478260 IC50 = 30 nM T31946 CMRO51 22478297 IC50 = 40 nM T31946 COB60M 23133320 IC50 = 50 nM T31946 C9QLP0 23133323 IC50 = 60 nM T31946 CQHK69 23646624 IC50 = 100 nM T31946 CC67EN 44405964 IC50 = 3200 nM T31946 CAVE92 44406020 IC50 = 14700 nM T31946 CJW6L4 44406041 IC50 = 1900 nM T31946 CTPE63 44406049 IC50 = 4100 nM T31946 C7Y9WO 46905535 IC50 > 15000 nM T31946 CB5O0I 49860186 IC50 = 30 nM T31946 C9W6SO 49860190 IC50 = 30 nM T31946 CLH49Z 59790029 IC50 = 2 nM T31946 C9QRX3 60098131 IC50 = 30 nM T31946 CV21FR 73349643 IC50 = 60 nM T31946 C9TMA1 73352657 IC50 = 8 nM T31946 CYQ8K1 73357210 IC50 = 3 nM T31946 C4AHL2 118711367 IC50 > 10000 nM T31946 C3K8AZ 135418423 IC50 = 320 nM T31946 CG1R7B 136087060 IC50 > 10000 nM T31946 CTA34O 145979089 IC50 = 276 nM T31946 D03HQK 5329843 IC50 = 14400 nM T31946 D03OKV 9844320 IC50 > 1000 nM T31946 D05THI 11174891 IC50 = 14000 nM T31946 D07XBW 9968373 IC50 = 530 nM T31946 D09LEK 5329850 IC50 = 4660 nM T31946 D09LKM 5329468 IC50 = 387 nM T31946 D09MSA 837182 IC50 = 6300 nM T31946 D0BM4F 5329404 IC50 = 3000 nM T31946 D0C6KI 5329006 IC50 = 1000 nM T31946 D0C6OD 11439243 IC50 = 11000 nM T31946 D0D3YL 5329849 IC50 = 1700 nM T31946 D0E3HC 5329450 IC50 = 18 nM T31946 D0M2QA 11245786 IC50 = 15000 nM T31946 D0UZ5W 975893 IC50 = 14000 nM T31946 D0V4BR 11266872 IC50 = 15000 nM T31946 D0V9DQ 5329847 IC50 = 1650 nM T31946 D0YN1E 5329454 IC50 = 622 nM T31946 D0YZ7H 9797370 IC50 = 3100 nM T04741 D0SV8E 126941 IC50 > 20000 nM T04741 D06YIB 135436405 IC50 = 130000 nM T04741 C7OTP8 3439 IC50 > 30000 nM T04741 CGZ59Q 65110 IC50 = 25000 nM T04741 CPY1X9 66546 IC50 = 7600 nM T04741 C6WED9 95887 IC50 = 54700 nM T04741 CF1M8Q 468708 IC50 > 30000 nM T04741 C14UVO 973584 IC50 = 34800 nM T04741 CT87OI 7033676 IC50 > 100000 nM T04741 CPQ64B 11227506 Ki = 3100 nM T04741 CHKA59 11963491 Ki = 230 nM T04741 CHB34X 11963492 Ki = 150 nM T04741 CBU8F6 12413165 Ki = 130 nM T04741 CPUO46 18084678 IC50 = 90000 nM T04741 CFV56S 44401945 Ki = 8000 nM T04741 CQP84U 44421387 IC50 = 36100 nM T04741 C3AYO8 44421389 IC50 = 203700 nM T04741 CDEA10 121378537 EC50 = 27 nM T04741 CFK7R6 121378562 EC50 = 17 nM T04741 CL3HE7 121378565 IC50 = 13 nM T04741 C1QVE3 121378588 EC50 = 7.6 nM T04741 CDS7C4 121378614 EC50 = 4 nM T04741 CA5FM9 121378618 EC50 = 31 nM T04741 CQFE10 121378639 EC50 = 7.9 nM T04741 CFPO56 121378656 IC50 = 14 nM T04741 C30WVM 121384725 EC50 = 18 nM T04741 C9ITU5 121384727 IC50 = 26 nM T04741 CPM86T 130297617 IC50 < 5 nM T04741 C9EA3J 135407589 IC50 = 700 nM T04741 CUS5Q1 135413518 Ki > 100000 nM T04741 CV46BA 135465343 Ki = 46000 nM T04741 CS0I8R 135469335 IC50 > 95000 nM T04741 CV47OY 135474781 Ki > 100000 nM T04741 CY5VG1 135488901 Ki = 8 nM T04741 C2R9FW 135491785 Ki > 100000 nM T04741 CVH8Q5 135502217 IC50 = 6400 nM T04741 CHD01N 135513031 Ki > 100000 nM T04741 CCF8H5 135545819 IC50 = 17000 nM T04741 CL2AG7 135566721 Ki > 100000 nM T04741 CRA6Z7 135566722 Ki > 100000 nM T04741 C06IDH 135746097 IC50 > 60000 nM T04741 CK7JZ1 135783338 IC50 = 3300 nM T04741 CH1W2S 135887126 IC50 = 62800 nM T04741 C6U0PF 135887127 IC50 = 141000 nM T04741 COA6S0 135887128 IC50 = 49900 nM T04741 CFIG79 135887147 IC50 > 100000 nM T04741 CDA05G 135887148 IC50 = 100000 nM T04741 CLBO26 135924167 Ki > 100000 nM T04741 C8R1PU 135924168 Ki > 100000 nM T04741 CN7B0Z 135924169 Ki > 100000 nM T04741 CYI9Q7 135924170 Ki = 20000 nM T04741 C5JDL6 135924171 Ki > 100000 nM T04741 C2SI7N 136002209 Ki = 17000 nM T04741 CRYC07 136002210 Ki = 52000 nM T04741 C6HL7E 136044121 IC50 > 40000 nM T04741 C76AYL 136044122 IC50 = 20000 nM T04741 C6F9VM 136044123 IC50 > 20000 nM T04741 CLFH92 136044127 IC50 = 20000 nM T04741 CQZ3T0 136044129 IC50 = 20000 nM T04741 CT0NK9 136046104 IC50 > 40000 nM T04741 CNW2I3 136117105 Ki = 6 nM T04741 CW6Y0D 136152909 Ki > 100000 nM T04741 C6MJY8 137647297 EC50 = 1811 nM T04741 CK4IQ7 137651195 IC50 = 18100 nM T04741 CHG9A5 137651614 IC50 < 5 nM T04741 C7LA3U 137653705 EC50 = 567 nM T04741 D02HXC 232556 Ki = 154 nM T04741 D03NSJ 413225 IC50 = 11600 nM T04741 D04JWS 324974 IC50 = 8800 nM T04741 D09KUE 259210 IC50 = 13900 nM T04741 D0A2JV 231116 IC50 = 16900 nM T04741 D0B3XP 235593 IC50 = 4100 nM T04741 D0F2WA 135929093 Ki > 100000 nM T04741 D0I2DB 235538 IC50 = 7800 nM T04741 D0R7LQ 135884475 Ki = 20000 nM T04741 D0S4MN 6280 IC50 = 231300 nM T04741 D0X2NH 44421368 IC50 = 9600 nM T04741 D0Z5WG 166760 Ki = 400 nM T00852 D03LWG 53235510 IC50 > 10000 nM T00852 D07HPJ 11476171 IC50 > 10000 nM T00852 D0K0YC 9826528 IC50 > 25000 nM T00852 C63WLY 89644 IC50 > 10 ug.mL-1 T00852 C5JE2Z 104860 IC50 = 5.5 ug.mL-1 T00852 CI1NA5 159926 IC50 = 7.7 ug.mL-1 T00852 CYBA43 177458 IC50 = 7.3 ug.mL-1 T00852 C8DX5E 4962846 IC50 = 4800 nM T00852 CDQ3M7 5359485 IC50 = 8 ug.mL-1 T00852 C54BYP 5360741 IC50 = 2.6 ug.mL-1 T00852 CBGE59 9833337 IC50 = 4800 nM T00852 CB6PJ8 9946185 IC50 > 50000 nM T00852 CG0V1T 11058385 IC50 = 940 nM T00852 CEXJ12 11186664 IC50 > 100000 nM T00852 CKR59O 11304151 IC50 = 800 nM T00852 CRTG16 11359538 IC50 > 20000 nM T00852 CT9V3D 11496376 IC50 = 2 nM T00852 C7HMO6 11526786 IC50 > 40000 nM T00852 CACS26 11561968 Ki > 4000 nM T00852 C1SW6R 11584834 IC50 = 28 nM T00852 C4GTZ8 11645322 IC50 > 20000 nM T00852 CU0E8O 11690457 Ki > 4000 nM T00852 CB0AP2 11705863 Ki > 4000 nM T00852 C4ZX9C 11989105 IC50 = 240 nM T00852 CDGF78 15282555 IC50 = 1600 nM T00852 CZHJ34 16058637 IC50 > 50000 nM T00852 CQW10N 16066845 IC50 = 19 nM T00852 CKX2L7 16085320 IC50 = 6 nM T00852 C8H3MQ 17758015 IC50 = 320 nM T00852 CA0C6P 17758017 IC50 = 41 nM T00852 CCFP63 17758018 IC50 = 43 nM T00852 C8AH1I 17758019 IC50 = 18 nM T00852 C1GKL6 17758020 IC50 = 20 nM T00852 C4OJ2C 17758135 IC50 = 910 nM T00852 CC7EN4 17758139 IC50 > 3000 nM T00852 C8S9VX 17758238 IC50 = 130 nM T00852 CIE58R 17758239 IC50 = 25 nM T00852 CO6LR5 17758240 IC50 = 20 nM T00852 CU0MF7 17758241 IC50 = 10 nM T00852 CME3S0 17758242 IC50 = 11300 nM T00852 CE73IF 17758353 IC50 = 20 nM T00852 CH9TR6 17758354 IC50 = 23 nM T00852 CWY3R6 17758355 IC50 = 830 nM T00852 CRMA95 17758356 IC50 > 5000 nM T00852 C2WA1B 17758357 IC50 = 250 nM T00852 CA79FH 17758358 IC50 = 16 nM T00852 CMOV50 17758462 IC50 = 500 nM T00852 CA7UV0 17758463 IC50 = 350 nM T00852 C29ZEO 17758464 IC50 = 2 nM T00852 CDRL71 17758465 IC50 = 110 nM T00852 CZK19Q 17758466 IC50 = 16 nM T00852 CKV5C8 17758467 IC50 = 16 nM T00852 CWH37T 17758574 IC50 = 30 nM T00852 C4NW2S 17758575 IC50 = 220 nM T00852 CA37KU 17758576 IC50 = 5900 nM T00852 CSA23C 17759556 IC50 = 160 nM T00852 C56YOG 17759673 IC50 = 130 nM T00852 CMG7F9 17759674 IC50 = 190 nM T00852 CIL8G9 17759675 IC50 = 130 nM T00852 CBC3V7 17759676 IC50 = 290 nM T00852 C60LUW 17759677 IC50 = 98 nM T00852 CGO0K1 17759678 IC50 = 280 nM T00852 CU90IN 17759786 IC50 = 170 nM T00852 C57NRL 17759787 IC50 = 18 nM T00852 CDER50 17759789 IC50 = 200 nM T00852 C5MXK8 17759790 IC50 = 87 nM T00852 CVHJ91 17759791 IC50 = 130 nM T00852 C1LAU8 18516243 IC50 = 710 nM T00852 CCPS81 24764502 IC50 > 35000 nM T00852 CJUK39 24770517 IC50 > 10000 nM T00852 C0EKO5 24772654 IC50 > 10000 nM T00852 C76HBA 24776415 IC50 = 130 nM T00852 CO5H7L 24776416 IC50 = 590 nM T00852 CE3WK7 24776417 IC50 = 220 nM T00852 C9PA0M 24807809 IC50 > 40000 nM T00852 CCP2M3 24822704 IC50 > 50000 nM T00852 C4V9GH 24894117 IC50 = 32000 nM T00852 CB5TP8 24894992 IC50 = 9600 nM T00852 CFW40U 24894997 IC50 = 40000 nM T00852 CN13JF 24899915 IC50 = 7.5 ug.mL-1 T00852 CBWR97 24899916 IC50 = 2.3 ug.mL-1 T00852 C9F2JD 24899917 IC50 > 10 ug.mL-1 T00852 C64MTI 24900160 IC50 = 9.7 ug.mL-1 T00852 CO2I6Q 24900161 IC50 > 10 ug.mL-1 T00852 CD5HQ0 24969301 IC50 > 10000 nM T00852 C4QF6H 25101222 IC50 = 10 nM T00852 CRO09K 25211064 IC50 > 40000 nM T00852 C8MBU1 25211459 IC50 = 560 nM T00852 CDET59 25218747 IC50 = 140 nM T00852 CFJ8E9 25218748 IC50 = 280 nM T00852 C8RGO1 25218749 IC50 = 210 nM T00852 CU96TR 25218750 IC50 = 50 nM T00852 C4X3EG 25218751 IC50 = 2900 nM T00852 C9SB8J 25218752 IC50 = 80 nM T00852 CV1K2M 25218753 IC50 = 310 nM T00852 CF9O0S 25218754 IC50 = 130 nM T00852 CKN8X4 25218755 IC50 = 20 nM T00852 C4T7YX 25218756 IC50 = 160 nM T00852 CJ5U1X 42639664 IC50 = 4.2 ug.mL-1 T00852 C48USC 44143344 IC50 = 1200 nM T00852 CUX7D9 44143345 IC50 = 40 nM T00852 CS53FU 44143346 IC50 = 170 nM T00852 CWBQ79 44143347 IC50 = 120 nM T00852 CE5CR9 44143348 IC50 = 140 nM T00852 CZ32DH 44143349 IC50 = 9.6 nM T00852 CP75VO 44143350 IC50 = 40 nM T00852 CNZ4U8 44143351 IC50 = 10 nM T00852 C7GP2Q 44143352 IC50 = 61 nM T00852 C6BP8W 44143353 IC50 = 40000 nM T00852 CS70WG 44143354 IC50 = 7 nM T00852 C6C8BM 44143355 IC50 = 23 nM T00852 C8Z9AV 44143356 IC50 = 20 nM T00852 CUDP56 44143357 IC50 = 4 nM T00852 CJ7Z5A 44143358 IC50 = 2 nM T00852 CZ4EK7 44143359 IC50 = 7.6 nM T00852 C5AGB3 44143360 IC50 = 3 nM T00852 C9Y2TI 44143361 IC50 = 17 nM T00852 C6K2OV 44143362 IC50 = 20 nM T00852 C7TQ0Z 44143363 IC50 = 13 nM T00852 C5ZD6S 44143364 IC50 = 22 nM T00852 C4YU9H 44143365 IC50 = 8 nM T00852 CPVM83 44143366 IC50 = 22 nM T00852 C1Z4BE 44143367 IC50 = 18 nM T00852 CH2OV4 44143368 IC50 = 5.3 nM T00852 CNDB53 44143369 IC50 = 2.2 nM T00852 C8YN5P 44143370 IC50 = 1.6 nM T00852 C9CWO1 44143371 IC50 = 8.2 nM T00852 C26XFL 44143372 IC50 = 9.1 nM T00852 C5SEQ2 44143373 IC50 = 10 nM T00852 C0VIX4 44219633 Ki > 4000 nM T00852 CWY0O8 44405398 IC50 = 21000 nM T00852 CLB87O 44405456 IC50 = 3400 nM T00852 CT0X5V 44405460 IC50 > 40000 nM T00852 C42RKW 44405465 IC50 > 40000 nM T00852 CRD42N 44405470 IC50 = 414 nM T00852 CC4ES0 44405474 IC50 > 40000 nM T00852 C0J4HD 44405491 IC50 = 140 nM T00852 CA06UN 44405502 IC50 > 40000 nM T00852 C5D4ZU 44405503 IC50 = 10000 nM T00852 CZ4VX0 44405504 IC50 = 380 nM T00852 CN69LX 44405505 IC50 > 40000 nM T00852 CZ4QD8 44405508 IC50 = 4600 nM T00852 CW18ZN 44405509 IC50 = 1800 nM T00852 CXK2D1 44405511 IC50 = 27000 nM T00852 C6V0UL 44405512 IC50 = 12 nM T00852 C02TLF 44405531 IC50 = 10000 nM T00852 CE4VU5 44405533 IC50 > 40000 nM T00852 CGM9Y5 44405534 IC50 = 4200 nM T00852 CUM6Z0 44405571 IC50 > 40000 nM T00852 C37LHW 44405576 IC50 > 40000 nM T00852 CA45EO 44405577 IC50 = 3565 nM T00852 CGI5L7 44405938 IC50 > 20000 nM T00852 C0G3WF 44405939 IC50 > 20000 nM T00852 CR3Q7Z 44405940 IC50 > 20000 nM T00852 C79WRL 44405941 IC50 > 20000 nM T00852 C0XZ8K 44406013 IC50 > 20000 nM T00852 CS3K1P 44406014 IC50 > 20000 nM T00852 CC93JP 44406018 IC50 > 20000 nM T00852 CCRZ12 44406074 IC50 > 20000 nM T00852 CF5R7J 44420059 IC50 = 640 nM T00852 C9M8KB 44420060 IC50 = 200 nM T00852 C4D9JC 44420064 IC50 = 210 nM T00852 CA2F6N 44420065 IC50 > 10000 nM T00852 C0IVY7 44420066 IC50 = 260 nM T00852 CBI78Z 44420071 IC50 > 40000 nM T00852 CWL94T 44420072 IC50 = 11000 nM T00852 C7HR9N 44420073 IC50 = 14 nM T00852 CQ4IL0 44420074 IC50 > 40000 nM T00852 C1IAH5 44420078 IC50 = 11500 nM T00852 C3C5YJ 44420079 IC50 = 60 nM T00852 CCNI18 44420080 IC50 > 40000 nM T00852 C6MEZ1 44420081 IC50 > 40000 nM T00852 CTNH25 44420086 IC50 = 100 nM T00852 C59FQZ 44420087 IC50 = 140 nM T00852 CZSY26 44420088 IC50 = 9200 nM T00852 CY3U0C 44420089 IC50 = 19000 nM T00852 CPAC82 44420091 IC50 = 110 nM T00852 CR5LE9 44420092 IC50 > 40000 nM T00852 CBJ20Y 44420096 IC50 = 31 nM T00852 CA45VH 44420104 IC50 = 74 nM T00852 CIYZ35 44420110 IC50 = 110 nM T00852 C0NFA3 44420116 IC50 = 2200 nM T00852 CUQ5V8 44420119 IC50 = 130 nM T00852 CP67UJ 44420120 IC50 = 90 nM T00852 CJPA07 44420123 IC50 = 30000 nM T00852 CO24YK 44420127 IC50 = 1000 nM T00852 CS7WT3 44420129 IC50 = 180 nM T00852 C0P4LG 44420135 IC50 > 40000 nM T00852 CSVU41 44420136 IC50 = 7000 nM T00852 CQ10XB 44420141 IC50 > 40000 nM T00852 CN58PE 44420142 IC50 > 10000 nM T00852 CNV92Z 44420143 IC50 = 3 nM T00852 CBIN31 44420144 IC50 = 3 nM T00852 CSA12W 44450544 IC50 = 50 nM T00852 CZI8O2 44580056 IC50 = 150 nM T00852 C4YOF5 44580057 IC50 = 120 nM T00852 CQL65I 44580058 IC50 = 170 nM T00852 CV0WF3 44580059 IC50 = 230 nM T00852 CM7DC1 44580107 IC50 = 50 nM T00852 C5JMS7 44580231 IC50 = 40 nM T00852 CHK18Y 44580626 IC50 > 50000 nM T00852 C6KBI0 44580627 IC50 > 50000 nM T00852 CK8C6W 44580674 IC50 = 410 nM T00852 CQ5M9I 44580675 IC50 = 540 nM T00852 CR8UE1 44580676 IC50 = 2200 nM T00852 CY4OE0 44580677 IC50 = 15000 nM T00852 CBS9W7 44580678 IC50 = 1700 nM T00852 C1Q8FZ 44580715 IC50 = 7500 nM T00852 C42ZJQ 44580716 IC50 = 1600 nM T00852 CL03FM 44580717 IC50 = 610 nM T00852 CEKG17 44580755 IC50 = 320 nM T00852 CX7E6T 44580756 IC50 = 90 nM T00852 C5V3PQ 44580757 IC50 = 310 nM T00852 CXNQ42 44580758 IC50 = 240 nM T00852 CR9LU0 44580759 IC50 = 130 nM T00852 CY3HW5 46224684 IC50 > 10000 nM T00852 C2P9QO 46228508 IC50 > 10000 nM T00852 C6E5PY 46228822 IC50 > 10000 nM T00852 C3T8AM 46228951 IC50 > 10000 nM T00852 CEQN27 52936621 Ki > 1000 nM T00852 CE06CY 53484072 IC50 = 180 nM T00852 C7NH2E 53484073 IC50 = 1000 nM T00852 CF13LC 56658822 IC50 > 100000 nM T00852 C27VAF 56662163 IC50 = 8100 nM T00852 CS6XU3 56662164 IC50 = 1700 nM T00852 CAI8L3 56662165 IC50 = 1700 nM T00852 CC2I1X 56662166 IC50 > 100000 nM T00852 C9N8KB 56662167 IC50 = 7100 nM T00852 C1MQC2 56662168 IC50 = 5100 nM T00852 CDY5U1 56662169 IC50 = 18000 nM T00852 C7X0NR 56665621 IC50 = 1200 nM T00852 CXJO92 56665622 IC50 > 100000 nM T00852 CJC2W0 56665623 IC50 > 100000 nM T00852 CJ1K5T 56665750 IC50 = 10000 nM T00852 CCT7G3 56669079 IC50 = 1100 nM T00852 CUK84P 56669080 IC50 = 22000 nM T00852 C7CLZ0 56669206 IC50 > 100000 nM T00852 C2Y6DO 56672540 IC50 = 3500 nM T00852 CDTF81 56672666 IC50 = 34000 nM T00852 CINZ90 56675920 IC50 = 34000 nM T00852 C07JAG 56675921 IC50 = 1500 nM T00852 C41CLO 56676036 IC50 = 6200 nM T00852 CCD7T8 56682544 IC50 > 100000 nM T00852 C9H8YW 56682660 IC50 = 2300 nM T00852 C2P8WS 56682661 IC50 > 100000 nM T00852 COH62U 60097413 IC50 > 4000 nM T00852 C1MR8Q 60097495 IC50 > 4000 nM T00852 C1HSE0 67035086 IC50 > 10000 nM T00852 CWI6K5 67035106 IC50 > 10000 nM T00852 C38RGB 67035556 IC50 > 10000 nM T00852 CV63UL 67240318 IC50 > 10000 nM T00852 C8I7GC 68293638 IC50 > 10000 nM T00852 CD56XK 68293660 IC50 > 10000 nM T00852 C5DGR9 69036886 IC50 = 1262 nM T00852 C3KLI5 118723185 IC50 > 100000 nM T00852 CAM6E1 121493969 IC50 = 270 nM T00852 CU17MH 132587462 IC50 = 4 nM T00852 CM2US4 134131972 IC50 = 200 nM T00852 C0QG8O 134132084 IC50 = 1300 nM T00852 C0TA9U 134132267 IC50 = 20 nM T00852 CGF13I 134132676 IC50 = 96 nM T00852 C09OLE 134135000 IC50 > 10000 nM T00852 CK35DH 134136236 IC50 = 600 nM T00852 CCS60I 134139857 IC50 = 90 nM T00852 CA65ZD 134140223 IC50 = 290 nM T00852 C40MWY 134140620 IC50 = 1010 nM T00852 C7E0UX 134141902 IC50 = 2600 nM T00852 CN3LB5 134142091 IC50 = 150 nM T00852 C91OZB 134144475 IC50 = 160 nM T00852 C8JVS6 134146432 IC50 = 38 nM T00852 CEA7V6 134148617 IC50 = 50 nM T00852 CO50GT 134149230 IC50 = 6 nM T00852 CQ2AR1 134149275 IC50 = 80 nM T00852 C27DEA 134149676 IC50 = 670 nM T00852 CH0K4X 134150907 IC50 = 100 nM T00852 CG34IL 134156318 IC50 = 1300 nM T00852 CT30MP 134156928 IC50 = 40 nM T00852 CQY20T 134157715 IC50 = 3500 nM T00852 C2AN7T 134611886 IC50 > 100000 nM T00852 CTIK72 135433080 IC50 = 47 nM T00852 CQE82W 135433128 IC50 > 100000 nM T00852 CC84EK 135454812 IC50 = 25000 nM T00852 CK2U1W 135484456 IC50 > 100000 nM T00852 CG5B2Y 135486151 IC50 > 100000 nM T00852 CTFQ18 135507472 IC50 = 38000 nM T00852 C1C0TF 135527102 IC50 = 109 nM T00852 CGC3Z6 135532406 IC50 > 100000 nM T00852 C9D0VX 135540521 IC50 = 4500 nM T00852 C6RI8B 135685743 IC50 = 16000 nM T00852 CX4ZB3 135863110 IC50 > 4000 nM T00852 CZO04G 135992153 IC50 = 18700 nM T00852 CA3MY1 135992306 IC50 = 3000 nM T00852 CZ6LK4 136019499 IC50 = 3200 nM T00852 C1GKH8 136025852 IC50 = 1126 nM T00852 C3BV9O 136025857 IC50 = 240 nM T00852 CE6U4P 136025998 IC50 = 10280 nM T00852 CWUZ51 136027078 IC50 = 1120 nM T00852 CLA7O9 136086929 IC50 = 418 nM T00852 C2OE7N 136086930 IC50 = 1734 nM T00852 CJ8P2B 136086931 IC50 = 1995 nM T00852 C7HKB5 136086932 IC50 = 1460 nM T00852 C9EGO6 136086933 IC50 = 2669 nM T00852 CCLH42 136086934 IC50 = 4943 nM T00852 C6FZ8O 136086935 IC50 = 20690 nM T00852 CDT46F 136086936 IC50 = 21395 nM T00852 CU3XK1 136086937 IC50 = 28300 nM T00852 C4ST6U 136086938 IC50 = 9260 nM T00852 CXC20K 136086939 IC50 > 100000 nM T00852 D03MUZ 17759555 IC50 = 12 nM T00852 D06HVH 54613583 IC50 > 10000 nM T00852 D06KSF 9549300 IC50 = 50 nM T00852 D06QWO 14824655 IC50 > 10 ug.mL-1 T00852 D06WGX 9549184 IC50 > 25000 nM T00852 D0A1CM 5281855 IC50 = 2370 nM T00852 D0F0AU 44405988 IC50 > 20000 nM T00852 D0G3SZ 6918469 IC50 = 8.8 ug.mL-1 T00852 D0J3LR 11634725 Ki > 4000 nM T00852 D0M5FF 5083 IC50 = 9950 nM T00852 D0V0QJ 389898 IC50 = 50 nM T43289 CGN48U 9827867 IC50 = 790 nM T43289 CW1G9B 10672666 IC50 > 10000 nM T43289 CW7Q2U 10895700 IC50 > 10000 nM T43289 CIQH43 11445130 IC50 = 1160 nM T43289 C37MRI 16718808 IC50 = 170 nM T43289 CVO5L6 24748791 IC50 = 5000 nM T43289 CS9TK6 38335241 IC50 > 10000 nM T43289 C30CFX 44436704 IC50 = 125 nM T43289 C78DJQ 71711730 IC50 < 10000 nM T43289 CM83VP 72163524 IC50 > 10000 nM T43289 CWP85J 87360663 IC50 > 10000 nM T43289 CJ6DA9 127028140 IC50 = 1440 nM T43289 CD9KI3 127028141 IC50 = 170 nM T43289 CW9NJ0 134415778 IC50 = 210 nM T43289 CUZ35A 138115400 IC50 = 794.33 nM T43289 CZR36C 155511554 IC50 = 199.53 nM T43289 C6NX4K 155519661 IC50 = 25.12 nM T43289 C4MS1B 155519676 IC50 = 12589.25 nM T43289 CN3BH5 155527998 IC50 = 1584.89 nM T43289 CHYW65 155528639 IC50 = 251.19 nM T43289 CD7O2G 155530095 IC50 = 7943.28 nM T43289 C35QWO 155531023 IC50 = 31.62 nM T43289 C12HON 155536142 IC50 = 1995.26 nM T43289 CY6DK3 155540964 IC50 = 100 nM T43289 C5MB9R 155547962 IC50 = 251.19 nM T43289 CLFB25 155548371 IC50 = 10000 nM T43289 COM52R 155551892 IC50 = 316.23 nM T43289 CJ3FI5 155553630 IC50 = 12589.25 nM T43289 CSW48V 155557718 IC50 = 6.31 nM T43289 CM8XB1 155565537 IC50 = 398.11 nM T43289 D0Y5IQ 44255320 IC50 = 10000 nM T31406 D09XZB 123631 IC50 = 110 nM T31406 D0E6XR 3062316 IC50 < 1 nM T31406 D0OB0F 5328940 IC50 = 3.2 nM T31406 D0R0MW 5329102 IC50 = 190 nM T31406 D0W5HK 216239 IC50 = 530 nM T31406 D03LWG 53235510 IC50 > 10000 nM T31406 D07EHV 44814409 IC50 > 10000 nM T31406 D0A5HC 45109868 IC50 = 52 nM T31406 D0E3TC 44259 IC50 = 1.9 nM T31406 D0M9QZ 11485656 IC50 > 50000 nM T31406 D03BNU 59604787 IC50 > 10000 nM T31406 D09HEV 6539952 IC50 = 0.4 nM T31406 D0T3ME 156422 IC50 = 1700 nM T31406 CBPM40 4878 IC50 = 5 nM T31406 C3W0JR 11379 EC50 > 1000000 nM T31406 C3R5VW 9547983 IC50 = 46 nM T31406 CV4J6S 9806451 IC50 = 3.467 nM T31406 CDTQ07 9870993 IC50 = 0.257 nM T31406 CYW49X 9927718 IC50 = 310 nM T31406 CCE2T5 10229750 IC50 = 901 nM T31406 C7SFI1 10296883 IC50 > 10000 nM T31406 CV1WZ5 10301047 IC50 = 4937 nM T31406 COE34F 11103319 IC50 > 19000 nM T31406 CD9E2W 11188787 IC50 = 8 nM T31406 CVOW82 11238420 IC50 = 10000 nM T31406 C25ZCN 11374110 IC50 > 50000 nM T31406 CREQ51 11429654 IC50 > 50000 nM T31406 CY0A4E 11429729 IC50 > 50000 nM T31406 CACS26 11561968 Ki > 2000 nM T31406 C9XI8Z 11574885 IC50 = 342 nM T31406 CA2KX0 11590078 IC50 > 50000 nM T31406 C1AUX0 11661290 IC50 = 85 nM T31406 CU0E8O 11690457 Ki > 2000 nM T31406 CE0KI4 11753519 IC50 = 20100 nM T31406 COFI19 11974316 IC50 = 456 nM T31406 C0M7TW 15948947 IC50 = 904 nM T31406 C1VNB4 15948949 IC50 = 27 nM T31406 CH8ZG5 15949048 IC50 = 16 nM T31406 CK2Z6Y 15949521 IC50 = 245 nM T31406 CBZF29 15949522 IC50 = 475 nM T31406 C34MCY 15949523 IC50 = 20 nM T31406 CS3P9G 15949524 IC50 = 9 nM T31406 C1KPH2 15949525 IC50 = 3826 nM T31406 C5JG9R 15949617 IC50 = 84 nM T31406 C8FT6U 15949618 IC50 = 844 nM T31406 C30PVQ 15949619 IC50 = 446 nM T31406 C3PNO2 15949620 IC50 = 11 nM T31406 C4I5RS 15949621 IC50 > 2500 nM T31406 CAIN63 15949888 IC50 > 2500 nM T31406 C2VDI1 15949889 IC50 = 192 nM T31406 COC02T 15949890 IC50 > 2500 nM T31406 CFQ6X3 15949974 IC50 = 69 nM T31406 CMKZ23 15949975 IC50 = 378 nM T31406 CWM5L4 15949976 IC50 = 31 nM T31406 CO7NG2 15950141 IC50 = 430 nM T31406 COIG45 15950224 IC50 = 43 nM T31406 C9V0TO 15950311 IC50 > 2500 nM T31406 CN36QI 16043219 IC50 = 48 nM T31406 CP3HS4 16220354 IC50 > 50000 nM T31406 CDZ31W 16747696 IC50 > 50000 nM T31406 CA7T2W 18450829 IC50 = 1410 nM T31406 CB2LF3 18450830 IC50 > 50000 nM T31406 CW0U4Z 18450843 IC50 = 1970 nM T31406 C6E4YZ 18450934 IC50 > 50000 nM T31406 C0VWB3 18451020 IC50 = 5970 nM T31406 C3J5HU 18451023 IC50 > 50000 nM T31406 CJA0D6 18451024 IC50 = 24200 nM T31406 C0X9RC 18451029 IC50 = 8800 nM T31406 CNBP94 18451030 IC50 = 21900 nM T31406 C6FQB7 18451036 IC50 = 13600 nM T31406 CEI23S 18451044 IC50 = 2360 nM T31406 CUZ1E0 18451049 IC50 = 4300 nM T31406 CGT10H 18451102 IC50 > 50000 nM T31406 CM9BN5 18451119 IC50 = 12900 nM T31406 CM1X8S 18451204 IC50 > 50000 nM T31406 CB84DI 18451225 IC50 = 45290 nM T31406 CYJ3M1 18451394 IC50 = 2360 nM T31406 C5ONK2 22736361 IC50 = 31 nM T31406 C7YG1N 24759534 IC50 = 30 nM T31406 CAJ4T2 24762205 IC50 = 181 nM T31406 C2UOE0 24766030 IC50 = 26 nM T31406 CS82HN 24856408 IC50 = 349 nM T31406 CZ5Y4H 24856498 IC50 = 456 nM T31406 CC10FW 24857629 IC50 = 215 nM T31406 CB79YC 24905143 IC50 = 23 nM T31406 C2DC9J 24905144 IC50 = 260 nM T31406 CN6V8Z 24905145 IC50 = 4 nM T31406 CSB7P5 24905148 IC50 = 8900 nM T31406 CGSF21 24905149 IC50 > 50000 nM T31406 CVDG02 24905150 IC50 < 1 nM T31406 CWH6C5 24905152 IC50 = 88 nM T31406 C0HE2Q 24905153 IC50 = 130 nM T31406 C7QSC9 24905154 IC50 = 2400 nM T31406 CO9D0K 24905155 IC50 = 1400 nM T31406 C5W9UR 24905157 IC50 = 7900 nM T31406 CC1DA3 24905158 IC50 = 4400 nM T31406 COW79F 24905159 IC50 = 3600 nM T31406 CFPA53 24905160 IC50 = 50000 nM T31406 C2O0JX 24905161 IC50 = 2300 nM T31406 CA72BE 24905162 IC50 = 5300 nM T31406 CQN6X9 24905163 IC50 = 12000 nM T31406 CD4O1F 24905165 IC50 = 1300 nM T31406 CKL48T 24905166 IC50 = 510 nM T31406 C76VYL 24905167 IC50 = 5000 nM T31406 C7K5PU 24905168 IC50 = 380 nM T31406 CZ57ID 24905169 IC50 = 180 nM T31406 C2DHX9 24905170 IC50 = 9200 nM T31406 CSB96E 24905171 IC50 = 13000 nM T31406 CWZ0R2 24905172 IC50 = 1000 nM T31406 CY3B6M 24905175 IC50 = 37 nM T31406 CW7UA3 24905176 IC50 = 113 nM T31406 CW1V0H 24905177 IC50 = 96 nM T31406 CO6Y0L 24905178 IC50 = 733 nM T31406 C60NQW 24905179 IC50 = 1600 nM T31406 C4MO8B 24905180 IC50 = 76 nM T31406 COJI47 24905181 IC50 = 28 nM T31406 CS0B2C 24905182 IC50 = 4.4 nM T31406 C1H4BT 24905183 IC50 = 2 nM T31406 C4WHK9 24905184 IC50 = 436 nM T31406 C7Q4MZ 24905185 IC50 = 9 nM T31406 CS4IP1 24905186 IC50 = 10 nM T31406 C69QWO 24905187 IC50 = 48 nM T31406 C85ANB 24905188 IC50 = 15 nM T31406 CNHD75 24905189 IC50 = 117 nM T31406 C9JUO2 24905190 IC50 = 1200 nM T31406 CPR03K 24905191 IC50 = 57 nM T31406 CTAG19 24905193 IC50 = 5.4 nM T31406 C7VJM5 24905194 IC50 = 889 nM T31406 CEP1L3 24905195 IC50 = 91 nM T31406 CP68ZD 24905196 IC50 = 56 nM T31406 C8Z0RJ 24905197 IC50 = 82 nM T31406 CN9RT0 24905198 IC50 = 567 nM T31406 CHI78P 24905200 IC50 = 422 nM T31406 CO6PE8 24905201 IC50 = 18 nM T31406 CZ63HS 24905202 IC50 = 10 nM T31406 C2X0FC 24905203 IC50 = 30 nM T31406 C0WCE3 24905204 IC50 = 100000 nM T31406 CNK50B 24905205 IC50 = 540 nM T31406 C12DPB 24905206 IC50 = 37 nM T31406 C8N0RH 24905207 IC50 = 540 nM T31406 CYA5G2 24905208 IC50 = 2200 nM T31406 CDV2B4 24905209 IC50 = 220 nM T31406 CEFK68 24905210 IC50 = 420 nM T31406 CUFP12 24905211 IC50 = 326 nM T31406 C0JG8L 24905212 IC50 = 5 nM T31406 CQ13ZI 24905215 IC50 = 100000 nM T31406 C6VI8F 24905216 IC50 = 878 nM T31406 CXNH25 24905217 IC50 = 1800 nM T31406 C2PN9S 24905218 IC50 = 946 nM T31406 C9O2AL 24905219 IC50 = 16000 nM T31406 CIT7U8 24905220 IC50 = 1600 nM T31406 CMD26S 24905221 IC50 = 153 nM T31406 C4R8WC 24905222 IC50 = 148 nM T31406 C47SHA 24905223 IC50 = 53 nM T31406 C1DY2R 24905224 IC50 = 33 nM T31406 CS0XF9 24905225 IC50 = 12000 nM T31406 CG5VX2 24905226 IC50 = 2700 nM T31406 C57QEO 24905227 IC50 = 1100 nM T31406 C7CG5E 24905228 IC50 = 4300 nM T31406 CHP5D1 24905229 IC50 = 2500 nM T31406 CXP09S 24905230 IC50 = 1100 nM T31406 CY7XG1 24905231 IC50 = 17000 nM T31406 C7JFQ2 24905232 IC50 = 17000 nM T31406 C2JM1P 24905233 IC50 = 3400 nM T31406 CC3BF0 24905234 IC50 = 17000 nM T31406 CE57FI 24905235 IC50 = 516 nM T31406 CUP20O 24905236 IC50 = 1000 nM T31406 CLC6Q2 24905237 IC50 = 4300 nM T31406 C9M1GI 24905238 IC50 = 855 nM T31406 CVD72F 24905239 IC50 = 35 nM T31406 CK38IZ 24905240 IC50 = 708 nM T31406 CO2V5E 24905241 IC50 = 4800 nM T31406 CZBA19 24905244 IC50 = 76 nM T31406 CQ8OI1 24905246 IC50 = 100000 nM T31406 CIF2J5 24905251 IC50 = 37 nM T31406 CPTE58 24905252 IC50 = 46 nM T31406 CP50RD 24905280 IC50 = 9.2 nM T31406 CG13ZM 24905281 IC50 = 13 nM T31406 CF0S6X 24905282 IC50 = 551 nM T31406 C5HBL0 24905284 IC50 = 12700 nM T31406 C2Z5DN 24905285 IC50 = 78 nM T31406 CL6GH8 24905286 IC50 = 624 nM T31406 CKYO98 24905287 IC50 = 5.1 nM T31406 CRNQ65 24905288 IC50 = 18 nM T31406 COD7I5 24905289 IC50 = 19 nM T31406 C4LP7E 24905290 IC50 = 65 nM T31406 CE9JC2 24905291 IC50 = 794 nM T31406 C2GI1R 24905292 IC50 = 6000 nM T31406 CHW8C4 24905293 IC50 = 115 nM T31406 CQF0H1 24905294 IC50 = 18 nM T31406 CNO7X0 24905295 IC50 = 2 nM T31406 C5WRG7 24905296 IC50 = 285 nM T31406 CQ1S0U 24905297 IC50 = 3400 nM T31406 C4UES7 24905298 IC50 = 861 nM T31406 CMS69P 24905299 IC50 = 1130 nM T31406 CC0U5M 24905300 IC50 = 0.18 nM T31406 CW7X6S 24905301 IC50 = 1530 nM T31406 C97IQV 24905302 IC50 = 4.5 nM T31406 CSJ47V 24905303 IC50 = 862 nM T31406 CPN74C 24905304 IC50 = 328 nM T31406 C5CS3N 24905305 IC50 = 67 nM T31406 CK4XE9 24905307 IC50 = 596 nM T31406 CTU6Z3 24905308 IC50 = 714 nM T31406 C9SQX1 24905309 IC50 = 25 nM T31406 CM75JP 24905310 IC50 = 86 nM T31406 C9Q2BJ 24905311 IC50 = 311 nM T31406 C9VUA1 24905312 IC50 = 20 nM T31406 CU3RS1 24905313 IC50 = 1200 nM T31406 CYG3H2 24905314 IC50 = 42 nM T31406 CV5Q7O 24905315 IC50 = 5.7 nM T31406 C8SA3O 24905316 IC50 = 10 nM T31406 CI5MN3 24905317 IC50 = 8.8 nM T31406 CJ1P7K 24905318 IC50 = 8 nM T31406 C1T6YQ 24905319 IC50 = 21 nM T31406 CAU86X 24905320 IC50 = 51 nM T31406 C54ISY 24905321 IC50 = 161 nM T31406 C2GE5I 24905322 IC50 = 33 nM T31406 C8D6YK 24905323 IC50 = 1400 nM T31406 C5NZH9 24905324 IC50 = 194 nM T31406 C9D6JR 24905325 IC50 = 11 nM T31406 CLZT41 24905326 IC50 = 5.8 nM T31406 CW8FD3 24905327 IC50 = 30 nM T31406 CHB7A2 24905328 IC50 = 258 nM T31406 CA8EI3 24905329 IC50 = 71 nM T31406 CCQ0O7 24905330 IC50 = 440 nM T31406 CJ81AS 24905331 IC50 = 24 nM T31406 C8PW4H 24905332 IC50 = 8.9 nM T31406 C2Y5TF 24905333 IC50 = 12 nM T31406 CH9FL5 24905334 IC50 = 2000 nM T31406 C1S0PC 24905335 IC50 = 920 nM T31406 C8N9MV 24905336 IC50 = 34 nM T31406 C9E8BJ 24905338 IC50 = 1500 nM T31406 CX85AC 24905341 IC50 = 13000 nM T31406 CKZ80E 24905342 IC50 = 47 nM T31406 CO8SH1 24905343 IC50 = 1100 nM T31406 C7IZL6 24905344 IC50 = 2400 nM T31406 CLW80F 44160269 IC50 = 5500 nM T31406 CN8WB9 44189332 IC50 = 958 nM T31406 CK73NR 44219749 IC50 > 50000 nM T31406 C3Z7VW 44414581 IC50 = 160 nM T31406 C8ED2X 44414624 IC50 = 546 nM T31406 CBS5K2 44432304 IC50 > 50000 nM T31406 CFJX63 44432305 IC50 = 2550 nM T31406 C54URN 44432306 IC50 = 2260 nM T31406 C57FJN 44432307 IC50 = 1290 nM T31406 C0PHT6 44432309 IC50 > 50000 nM T31406 CGV37F 44440254 IC50 = 30270 nM T31406 C5JUV3 44440256 IC50 > 50000 nM T31406 CFB56S 44440259 IC50 > 50000 nM T31406 CEW9G2 44440261 IC50 > 50000 nM T31406 C4WRN5 44541014 IC50 = 27100 nM T31406 CJY8S0 44570884 IC50 > 5000 nM T31406 C28QLM 44605035 IC50 > 50000 nM T31406 C75XHS 44605037 IC50 > 50000 nM T31406 CVED60 45254198 IC50 = 197 nM T31406 C53MQJ 45254575 IC50 = 164 nM T31406 CS9Y8K 45254577 IC50 = 26 nM T31406 C7YCA2 45257074 IC50 = 208 nM T31406 C19HUI 45257075 IC50 = 187 nM T31406 CC95PQ 45375865 IC50 = 550 nM T31406 CEOQ27 45375866 IC50 > 50000 nM T31406 C96BNW 46179972 IC50 = 16 nM T31406 CZBL95 46220496 IC50 = 475 nM T31406 CX8MJ9 46836027 IC50 = 1117 nM T31406 CS8NX0 46836043 IC50 = 807 nM T31406 CO3P0J 46866604 IC50 < 50000 nM T31406 CX43UQ 46871756 IC50 = 310 nM T31406 CRS61F 46879438 IC50 > 2500 nM T31406 C27JEF 46879439 IC50 > 2500 nM T31406 CF0T8P 46879440 IC50 = 1810 nM T31406 C12RMW 46879441 IC50 > 2500 nM T31406 CH2D7N 46879442 IC50 = 1875 nM T31406 CI6OD8 46879443 IC50 = 56 nM T31406 C7YD4Q 46879444 IC50 = 130 nM T31406 C8MN5Q 46879445 IC50 = 260 nM T31406 CX6SW2 46879446 IC50 > 2500 nM T31406 CNF3V6 46879447 IC50 > 2500 nM T31406 CW46VY 46879448 IC50 = 54 nM T31406 CLK6X3 46879907 IC50 = 121 nM T31406 CRPU47 46879908 IC50 = 46 nM T31406 C1TIE9 46880013 IC50 > 2500 nM T31406 C2A8KO 46880066 IC50 > 2500 nM T31406 CBRP80 46880067 IC50 = 1960 nM T31406 C3FY2B 46880068 IC50 = 345 nM T31406 CX89TY 46880069 IC50 = 65 nM T31406 CB0XY1 46880070 IC50 = 49 nM T31406 CUD81V 46880071 IC50 = 805 nM T31406 CZP58Q 46880072 IC50 = 450 nM T31406 CC8OF9 46880073 IC50 = 917 nM T31406 CF41HG 46880098 IC50 = 405 nM T31406 C6O2YG 46880099 IC50 > 2500 nM T31406 CI78DM 46880100 IC50 = 151 nM T31406 CU04ZK 46880101 IC50 = 139 nM T31406 C4E0MF 46880133 IC50 > 2500 nM T31406 COJ16A 46880134 IC50 > 2500 nM T31406 C71MGJ 46880135 IC50 > 2500 nM T31406 CJOM49 46880136 IC50 = 1240 nM T31406 C3R6TL 46880213 IC50 > 2500 nM T31406 CT8BQ4 46880214 IC50 > 2500 nM T31406 C0JTO4 46880215 IC50 > 2500 nM T31406 CAFN49 46880216 IC50 > 2500 nM T31406 C1YS5A 46890918 IC50 > 1000 nM T31406 CJ5S3N 46890968 IC50 = 37 nM T31406 CAGE32 46890969 IC50 = 295 nM T31406 C3A7BP 46890970 IC50 = 594 nM T31406 CTV73J 46890971 IC50 = 193 nM T31406 CUX9B4 46891024 IC50 = 172 nM T31406 CG35WP 46891025 IC50 = 70 nM T31406 C3FBH0 46891026 IC50 = 110 nM T31406 CYOU90 46891080 IC50 = 14 nM T31406 CJ16KH 46891081 IC50 = 256 nM T31406 C7DOF4 46891082 IC50 = 88 nM T31406 CM14YO 46891147 IC50 = 21 nM T31406 CRPL41 46891148 IC50 = 178 nM T31406 C6FJ7G 46891184 IC50 > 1000 nM T31406 C1B2UZ 46891185 IC50 > 1000 nM T31406 CYM5B2 46891226 IC50 > 1000 nM T31406 C2DZE0 46891227 IC50 = 676 nM T31406 C1W0JX 46891228 IC50 = 270 nM T31406 CI3VZ0 46891275 IC50 > 1000 nM T31406 C46STW 51346068 Ki > 1250000 nM T31406 CEQN27 52936621 Ki > 1000 nM T31406 CU1P2L 52940797 IC50 = 10500 nM T31406 CDHJ08 52942235 IC50 = 7900 nM T31406 C1XEV2 52943394 IC50 = 244 nM T31406 CWPC54 52945348 IC50 = 270 nM T31406 C4NLX7 52945630 IC50 = 1200 nM T31406 CXD6T8 52945845 IC50 = 2300 nM T31406 C6DC4S 53241447 IC50 = 110 nM T31406 C8NA4L 53384644 IC50 > 30000 nM T31406 CP1FH5 53391990 IC50 = 51 nM T31406 C4JCT1 53476174 IC50 = 82 nM T31406 CBS73R 53484203 Ki = 1720 nM T31406 CAR67O 56665753 Ki = 3870 nM T31406 CLHO15 56676037 Ki = 5000 nM T31406 C6HR5F 58416745 IC50 = 829 nM T31406 CRY9K7 58416748 IC50 = 625 nM T31406 CYI32L 58532548 IC50 = 8552 nM T31406 CXJ63M 59603829 IC50 = 33 nM T31406 CQEU96 59603842 IC50 = 2.8 nM T31406 C1MR8Q 60097495 IC50 > 1000 nM T31406 CV63UL 67240318 IC50 > 10000 nM T31406 CAIO65 68796885 IC50 = 22 nM T31406 C5DGR9 69036886 IC50 = 1855 nM T31406 CDP96Z 69788774 IC50 = 15 nM T31406 CZM1K4 71765510 IC50 = 99 nM T31406 CI9H6L 72164895 Ki = 504 nM T31406 C3ZHD0 73051195 IC50 = 7.6 nM T31406 CTZJ26 73051657 IC50 = 13.49 nM T31406 C1HW4B 89735655 IC50 = 6400 nM T31406 CTH6D8 118105272 IC50 = 9 nM T31406 C0LCN1 118105340 IC50 = 3.7 nM T31406 CDYX60 118105350 IC50 = 90 nM T31406 CCXA46 122190499 Ki = 980 nM T31406 C3PQ4W 122190505 Ki = 730 nM T31406 CN1DK0 122190507 Ki = 1200 nM T31406 C2LAM7 126591927 IC50 = 137 nM T31406 C3NHU5 127030449 IC50 = 482 nM T31406 CI73JH 127030772 IC50 > 17000 nM T31406 CEI25F 127030791 IC50 = 3221 nM T31406 CUQ5T4 127030792 IC50 = 2141 nM T31406 C7Q6PH 127030793 IC50 = 13291 nM T31406 CRO3B9 127031107 IC50 > 16000 nM T31406 CXV6F2 127031108 IC50 > 15000 nM T31406 C90LYU 127031109 IC50 = 26 nM T31406 CD5A9R 127031117 IC50 = 692 nM T31406 CV7KB9 127031414 IC50 > 16000 nM T31406 CANH59 127031725 IC50 = 8673 nM T31406 C3UDF1 127034594 IC50 > 19000 nM T31406 C5H8OZ 131632969 IC50 = 1318.26 nM T31406 CZ8Q6N 131632970 IC50 = 208.93 nM T31406 C8DLX3 131632971 IC50 = 111 nM T31406 CO6N0Q 131632972 IC50 = 686 nM T31406 C6NQG3 131704413 IC50 = 10.96 nM T31406 C8I7HV 132602209 IC50 = 13 nM T31406 CU29YK 135750268 IC50 = 47 nM T31406 C12UDA 135947972 IC50 = 26 nM T31406 CN42ZS 135947973 IC50 = 23 nM T31406 CF8AO3 135947974 IC50 = 76 nM T31406 CW08GJ 135947976 IC50 = 248 nM T31406 CJN7E2 135947978 IC50 = 100 nM T31406 CFKH34 135947979 IC50 = 20 nM T31406 CXC69T 137321158 IC50 = 142 nM T31406 C28QUP 137652864 IC50 = 199.4 nM T31406 CU64FZ 145963919 IC50 = 52 nM T31406 CT9D0I 145964074 IC50 = 18 nM T31406 C9BNT0 145964156 IC50 = 27 nM T31406 CIT76X 145964368 IC50 = 65 nM T31406 CIL40C 145964733 IC50 = 7.4 nM T31406 C8J3AE 145965430 IC50 = 6.9 nM T31406 C8LF7A 145965583 IC50 = 119 nM T31406 CS8DW3 145965618 IC50 = 1.8 nM T31406 C4XJ7Z 145966726 IC50 = 36 nM T31406 CQO63F 145971860 IC50 = 7.5 nM T31406 CV6IX5 145972308 IC50 = 6.3 nM T31406 CF49ZG 145977457 IC50 = 5.4 nM T31406 CC2AQ0 154573782 IC50 = 3 nM T31406 C2MD1Q 155513187 IC50 > 10000 nM T31406 C3NA2I 155519537 IC50 = 33 nM T31406 C54ARD 155532371 IC50 > 100000 nM T31406 D03EHM 24905142 IC50 = 8 nM T31406 D03OKV 9844320 IC50 > 23 nM T31406 D06HVH 54613583 IC50 > 10000 nM T31406 D06WGX 9549184 IC50 = 1220 nM T31406 D08RZB 11153014 IC50 = 2 nM T31406 D0H2CM 135565635 IC50 = 1200 nM T31406 D0IR6U 5494425 IC50 = 7700 nM T62449 D0EG1I 9926791 IC50 > 10000 nM T62449 D0R0MW 5329102 IC50 = 77.27 nM T62449 D00NZL 11955855 IC50 = 10.4 nM T62449 D02RJY 11442891 IC50 > 10000 nM T62449 D03HUX 49792852 IC50 > 10000 nM T62449 D05FWH 46239015 IC50 = 3 nM T62449 D06KTJ 53252276 IC50 = 50 nM T62449 D08UUL 46700756 IC50 = 0.56 nM T62449 D09YDM 24360 EC50 = 2.1 nM T62449 D0A5MC 11712649 IC50 > 100000 nM T62449 D0E3TC 44259 IC50 < 0.1 nM T62449 D0O0LS 25141092 IC50 > 10000 nM T62449 D0P1CV 46191454 IC50 > 10000 nM T62449 D0PM7Q 11152667 IC50 = 5 nM T62449 D0Q7RE 16007391 Ki > 10000 nM T62449 D0Q9UX 16718576 IC50 > 10000 nM T62449 D0S5RC 3025986 IC50 > 40000 nM T62449 D0Z9VY 72271 IC50 = 9.88 nM T62449 D03BNU 59604787 IC50 > 3500 nM T62449 D0YK9D 9956119 IC50 > 10000 nM T62449 D0H4GI 10275001 IC50 > 3000 nM T62449 D0T3ME 156422 IC50 > 30000 nM T62449 C3J8HY 40118 Ki = 39810.72 nM T62449 C6S5PV 40119 Ki = 501.19 nM T62449 CM6C0O 70836 IC50 > 50000 nM T62449 C0KBL4 81900 Ki = 39810.72 nM T62449 CIB4U6 98614 IC50 = 52000 nM T62449 CM9GA6 290208 IC50 > 100000 nM T62449 C1ZG2U 449087 IC50 > 10000 nM T62449 CN47JV 665387 Ki = 3162.28 nM T62449 CP71KC 683649 IC50 = 1400 nM T62449 C49BUD 1417635 IC50 > 100000 nM T62449 CXQ3W7 1583275 IC50 > 100000 nM T62449 C4WFP1 1587957 Ki = 13700 nM T62449 CZL67G 1596636 IC50 > 100000 nM T62449 C1X3LF 2059510 Ki = 7200 nM T62449 C9ZT2G 2753118 Ki = 100000 nM T62449 CHC5I0 2971839 IC50 > 10000 nM T62449 CPOJ12 3078519 IC50 = 5.6 nM T62449 CK05YM 3653116 Ki = 15848.93 nM T62449 CR9LG3 4369432 IC50 = 6100 nM T62449 CTXC93 4369433 Ki = 1300 nM T62449 CU5B1Z 4369491 IC50 = 47 nM T62449 CG17TN 6914611 IC50 = 4200 nM T62449 C7E2QK 6914613 IC50 = 16000 nM T62449 C2PGU4 9572071 IC50 > 7900000 nM T62449 CA3V0T 9572240 IC50 > 100000 nM T62449 C1DJ6B 9572244 IC50 > 100000 nM T62449 C73SQF 9572245 IC50 > 100000 nM T62449 CJR60A 9572531 IC50 > 100000 nM T62449 C7GBL9 9572533 IC50 > 100000 nM T62449 C8P3DE 9572535 IC50 > 100000 nM T62449 C6MU5H 9572537 IC50 > 100000 nM T62449 CXZK43 9572545 IC50 > 100000 nM T62449 CDF2S5 9572547 IC50 > 100000 nM T62449 CXI68F 9572620 IC50 > 100000 nM T62449 CSG4X7 9572624 IC50 > 100000 nM T62449 CIFU15 9572626 IC50 > 100000 nM T62449 C7OZ6U 9572657 IC50 > 100000 nM T62449 CU30ZL 9572659 IC50 > 100000 nM T62449 C6NGW1 9572661 IC50 > 100000 nM T62449 CRA10N 9572663 IC50 > 100000 nM T62449 C7J4HC 9572736 IC50 > 100000 nM T62449 C5DX4K 9814559 IC50 = 5000 nM T62449 CN9T7I 9815578 IC50 = 800 nM T62449 C9H0PI 9844011 Ki = 19.95 nM T62449 CE15KX 9847909 IC50 = 24 nM T62449 CM5Z8X 9869943 IC50 > 1000 nM T62449 C0ZF8B 9878679 IC50 = 890 nM T62449 CY3AQ0 9902908 IC50 = 150 nM T62449 C6R5KY 9923895 IC50 = 1000 nM T62449 CJO47T 9948405 IC50 > 10000 nM T62449 CEI07F 9967283 IC50 = 110 nM T62449 CGW03A 9975362 IC50 = 4200 nM T62449 CHR0C2 9975831 Ki = 10 nM T62449 CWD27O 9976672 IC50 > 50000 nM T62449 CZ2F6K 9976901 IC50 = 480 nM T62449 CQ0SW7 9978312 IC50 = 410 nM T62449 CG4M8W 9980097 IC50 = 230 nM T62449 CPM0D4 9981170 IC50 = 3 nM T62449 C4XM8Q 9982874 Ki = 19.95 nM T62449 C7HK4S 9993058 IC50 = 40 nM T62449 CEP27R 9993745 IC50 = 30 nM T62449 CG7MA0 9997535 IC50 = 1600 nM T62449 CV8I5X 9999342 IC50 > 10000 nM T62449 CD1O6A 10000495 IC50 = 120 nM T62449 CLRN75 10001302 IC50 = 27000 nM T62449 CI63HK 10001419 IC50 = 420 nM T62449 COV18R 10003686 Ki = 6.31 nM T62449 C0XNP5 10005624 IC50 = 7000 nM T62449 C0UK4L 10008287 IC50 = 8000 nM T62449 CE63WU 10022438 IC50 = 220 nM T62449 C0GMQ1 10022580 IC50 = 1100 nM T62449 CZF32P 10022581 IC50 = 130 nM T62449 CUW08Y 10038490 IC50 = 1600 nM T62449 CCP9A1 10043931 IC50 = 500 nM T62449 C59IGN 10044928 IC50 = 53 nM T62449 CAZ8D2 10046459 IC50 = 35 nM T62449 CXVI60 10050866 Ki = 158.49 nM T62449 CV2Y8H 10051869 IC50 = 53 nM T62449 C6PXJ7 10065463 IC50 = 120 nM T62449 C9JB0D 10068075 IC50 = 15 nM T62449 CSY3B7 10071975 IC50 = 580 nM T62449 C7I9RE 10088687 IC50 = 33 nM T62449 C8PDE5 10089771 IC50 = 48 nM T62449 CQ4PS1 10091673 IC50 = 29 nM T62449 C3S8QE 10098139 IC50 = 2.8 nM T62449 CNZ28P 10098763 IC50 = 750 nM T62449 CJCX10 10109058 IC50 = 37 nM T62449 CU5ID6 10126538 IC50 = 3465 nM T62449 C8BGJ1 10126790 IC50 = 47 nM T62449 C5X4VI 10127458 IC50 = 75 nM T62449 CJ3B0R 10134310 IC50 = 4100 nM T62449 C5EQB2 10156987 IC50 = 140 nM T62449 C0PG4T 10172394 IC50 = 120 nM T62449 CB03KN 10173666 IC50 = 1280 nM T62449 CU1F3Q 10193410 IC50 = 2839 nM T62449 CTC89D 10194362 Ki = 3162.28 nM T62449 CQ63XF 10199113 Ki = 1995.26 nM T62449 CZ3H0I 10199486 IC50 = 23000 nM T62449 C0R5AX 10215912 IC50 = 4 nM T62449 C5CS7N 10221890 IC50 = 230 nM T62449 C5TQ7X 10247543 IC50 > 10000 nM T62449 CNCY43 10247868 IC50 = 88 nM T62449 CCQP92 10248686 IC50 = 88 nM T62449 CNQH37 10253652 IC50 = 1400 nM T62449 C2HF4M 10266513 IC50 = 60 nM T62449 C4C8WB 10287456 IC50 = 1306 nM T62449 CT4D7G 10309409 IC50 = 92 nM T62449 CVNL94 10310919 Ki = 125.89 nM T62449 CO8N7L 10318383 IC50 = 600 nM T62449 C3PV5R 10318616 IC50 = 240 nM T62449 C8C2TF 10319524 IC50 = 1300 nM T62449 C83YTG 10319891 IC50 = 35000 nM T62449 CDB7F4 10321590 IC50 = 450 nM T62449 C0QYU7 10333656 IC50 = 14 nM T62449 CX5K6W 10337485 IC50 = 790 nM T62449 CURW95 10337978 IC50 = 91 nM T62449 CF8C3S 10341125 IC50 = 6 nM T62449 C0A3KS 10342897 IC50 = 4400 nM T62449 C7I1GX 10343927 IC50 = 620 nM T62449 C3FS9T 10355488 IC50 = 30 nM T62449 CUO1G6 10359398 Ki = 79.43 nM T62449 CULF78 10362050 IC50 = 69 nM T62449 C1EYA2 10364585 IC50 = 18 nM T62449 C6G9VY 10369451 IC50 = 77 nM T62449 CHN1P0 10384072 IC50 = 440 nM T62449 C9NOZ2 10385019 IC50 = 790 nM T62449 C2G3DY 10386664 IC50 = 150 nM T62449 C0UJ5R 10389002 IC50 = 120 nM T62449 CP5IH6 10390085 IC50 = 630 nM T62449 CK4CE8 10405212 IC50 = 21 nM T62449 CZO8B1 10406209 Ki = 79.43 nM T62449 C84OIA 10406993 IC50 = 4000 nM T62449 CB7FK9 10407121 IC50 = 7.9 nM T62449 C2VR3A 10410783 IC50 = 77 nM T62449 C29BMY 10413815 IC50 = 1300 nM T62449 CEF98R 10413846 IC50 = 120 nM T62449 CH8KM7 10414039 IC50 = 2500 nM T62449 C6H9BL 10429435 IC50 = 7 nM T62449 C7HBP6 10429593 IC50 > 10000 nM T62449 CAU5M6 10430419 IC50 = 12 nM T62449 C5P1XN 10431859 IC50 = 2400 nM T62449 C7UI1E 10431917 IC50 > 50000 nM T62449 CO7Q6H 10434889 IC50 = 55 nM T62449 COP9B6 10435655 IC50 = 420 nM T62449 CR4B6L 10450912 IC50 > 10000 nM T62449 CGC12F 10451785 IC50 = 110 nM T62449 CE5HU9 10453390 IC50 = 1200 nM T62449 C4A9NC 10472653 IC50 = 1200 nM T62449 C2WQ8M 10473563 IC50 > 10000 nM T62449 CD25UL 10475362 IC50 = 5300 nM T62449 CJI7L5 10475450 IC50 = 15 nM T62449 CG9EZ5 10476278 Ki = 7.943 nM T62449 CC3DV9 10477305 IC50 = 220 nM T62449 CM5WA8 10478085 IC50 = 180 nM T62449 CV3HS7 11107024 IC50 > 50000 nM T62449 CE7S5B 11155895 IC50 = 63 nM T62449 CTLB14 11175629 IC50 = 34 nM T62449 CS59ZY 11185396 IC50 = 1.2 nM T62449 C98PNC 11187517 IC50 = 3 nM T62449 C7K4LR 11189930 IC50 = 26 nM T62449 CMG5O4 11200878 IC50 = 7 nM T62449 C9C6UP 11222364 IC50 = 37 nM T62449 COA0M5 11234350 EC50 = 30 nM T62449 C2FNL3 11234351 EC50 = 60 nM T62449 C4DI8W 11236121 IC50 > 100000 nM T62449 C95JDI 11236215 IC50 = 5 nM T62449 CC28NA 11236402 IC50 = 11 nM T62449 CN6Y9I 11249510 IC50 = 2 nM T62449 CF3L9O 11257518 IC50 = 19 nM T62449 CTD09Z 11268805 IC50 = 5 nM T62449 C84PYR 11291546 Ki = 15.85 nM T62449 CBOP58 11293798 IC50 = 2 nM T62449 C29IST 11302358 IC50 = 5500 nM T62449 C78QPV 11303495 IC50 = 14 nM T62449 C5RM8B 11304347 IC50 > 100000 nM T62449 CX3B6P 11304642 IC50 = 12 nM T62449 CK6IJ4 11305731 IC50 = 1 nM T62449 CHI42X 11306184 IC50 = 19 nM T62449 C30MLR 11313946 EC50 = 19 nM T62449 C1I9DH 11315248 IC50 = 3 nM T62449 CJEA47 11316746 IC50 = 17 nM T62449 CPQ6H1 11317619 IC50 = 9 nM T62449 C0RNS6 11329100 Ki = 12.59 nM T62449 CXLY64 11337725 IC50 = 10 nM T62449 C39RGW 11338178 IC50 = 10 nM T62449 CH0FO1 11338464 IC50 = 13 nM T62449 C65RFW 11339762 IC50 = 15 nM T62449 CZJ5O2 11339836 IC50 = 5 nM T62449 CY1OK7 11348631 Ki = 7.943 nM T62449 C8NSB7 11348767 IC50 = 8 nM T62449 CQ82SW 11349000 IC50 = 9 nM T62449 CN1SI8 11349961 IC50 = 69 nM T62449 CZX49R 11360110 IC50 = 15 nM T62449 CU2DS9 11360680 IC50 = 6 nM T62449 C2MSA4 11362027 IC50 = 12 nM T62449 C26BZX 11362471 Ki = 4.3 nM T62449 CCNM49 11363612 IC50 = 91 nM T62449 C43NPS 11373886 IC50 > 10000 nM T62449 C3DQO1 11385547 IC50 = 139 nM T62449 CH3ET6 11396653 IC50 = 248 nM T62449 CWXB93 11397177 Ki = 13.7 nM T62449 CGI54M 11397537 IC50 = 2 nM T62449 CWM18I 11406175 IC50 = 7 nM T62449 C72TPC 11416654 IC50 = 10 nM T62449 C1WXC5 11417488 IC50 = 8 nM T62449 CWLY42 11418927 IC50 = 10 nM T62449 C0APW4 11422034 IC50 > 10000 nM T62449 C60AYD 11428760 IC50 = 7 nM T62449 CA8W1F 11429573 IC50 = 2 nM T62449 CTY7L3 11430448 IC50 = 6 nM T62449 C8CA3E 11440353 EC50 = 10 nM T62449 CF1GA8 11440387 EC50 = 20 nM T62449 CV9E4I 11442872 IC50 = 1 nM T62449 CBNR79 11443264 IC50 = 9 nM T62449 C6HKS9 11451776 IC50 = 10 nM T62449 C3T9YB 11473431 IC50 > 100000 nM T62449 CDI94K 11473432 IC50 > 100000 nM T62449 CGMN46 11474470 EC50 = 60 nM T62449 CJG34W 11474546 IC50 = 39 nM T62449 CNR8J3 11485833 IC50 = 97 nM T62449 CRZL12 11488502 IC50 = 12 nM T62449 C0H6QS 11495680 IC50 > 10000 nM T62449 CIW9L5 11502867 IC50 > 10000 nM T62449 CK2Q0X 11516978 IC50 > 10000 nM T62449 COD7K5 11517939 IC50 = 100 nM T62449 CH3Q9P 11518244 IC50 = 10 nM T62449 CPE53F 11526238 IC50 > 10000 nM T62449 C5BM4T 11531799 IC50 > 10000 nM T62449 C53OSD 11532048 IC50 > 10000 nM T62449 CC4QM5 11532676 IC50 > 10000 nM T62449 CTG83F 11539329 Ki > 8800 nM T62449 C01FVM 11546457 IC50 > 10000 nM T62449 C2GKE5 11547522 IC50 = 50 nM T62449 CACS26 11561968 Ki > 2000 nM T62449 CNBM81 11562171 IC50 > 10000 nM T62449 CMIL86 11590363 Ki > 8800 nM T62449 C0NV9Y 11596881 IC50 > 10000 nM T62449 CC9WA7 11612456 IC50 = 5 nM T62449 C1BLZ5 11620055 IC50 > 10000 nM T62449 CA0O3I 11623420 IC50 = 2900 nM T62449 CSM62L 11626920 IC50 > 30000 nM T62449 C9T6SC 11640926 Ki > 8800 nM T62449 CI9L7G 11648145 IC50 = 100 nM T62449 C24GRQ 11661959 IC50 > 10000 nM T62449 CO4S7F 11662575 IC50 = 35 nM T62449 CV3HS2 11664426 Ki = 6.31 nM T62449 CU3I9Q 11676957 IC50 = 10 nM T62449 CS72ED 11682843 IC50 > 10000 nM T62449 CCME06 11690363 EC50 = 97 nM T62449 CU0E8O 11690457 Ki > 2000 nM T62449 CLC53E 11691173 IC50 > 10000 nM T62449 CERT40 11698764 IC50 = 6 nM T62449 CB0AP2 11705863 Ki > 10000 nM T62449 C1FTX3 11719305 IC50 > 10000 nM T62449 CY54HB 11722980 IC50 = 970 nM T62449 CO15FK 11725319 IC50 = 72 nM T62449 CLZU92 11739898 IC50 = 1400 nM T62449 CTSG65 11740347 IC50 = 230 nM T62449 CW4EK0 11740418 IC50 = 970 nM T62449 CAOB03 11744406 IC50 = 200 nM T62449 CE1N3Y 11744724 IC50 = 410 nM T62449 C27SQU 11749860 IC50 = 24 nM T62449 CI25FG 11751448 IC50 = 109 nM T62449 CPUL52 11774385 IC50 = 4 nM T62449 CT49SI 11774807 IC50 = 13 nM T62449 C6T0RG 11784520 IC50 = 3 nM T62449 C2CN8L 11784902 IC50 = 12 nM T62449 CG6Q1B 11842628 IC50 = 7 nM T62449 CU9RM0 11842834 IC50 = 38 nM T62449 CGSY90 11842835 IC50 > 10000 nM T62449 CZ23AN 11842836 IC50 = 210 nM T62449 CR25PH 11842837 IC50 = 430 nM T62449 CYHR74 11842838 IC50 = 370 nM T62449 C14TDN 11842839 IC50 > 10000 nM T62449 CVR2K9 11842841 IC50 = 7100 nM T62449 C1Z3RW 11842842 IC50 > 10000 nM T62449 CG3NR8 11842843 IC50 = 710 nM T62449 C05ALU 11842844 IC50 = 160 nM T62449 CL3Q1S 11842845 IC50 = 24000 nM T62449 CULN90 11842846 IC50 = 2300 nM T62449 CCG3Q9 11842994 IC50 > 10000 nM T62449 CUMC05 11842995 IC50 > 10000 nM T62449 C87DLM 11842996 IC50 > 10000 nM T62449 CQ6H1Z 11842997 IC50 = 77 nM T62449 CKDH12 11842998 IC50 = 19000 nM T62449 C2EXY1 11842999 IC50 = 450 nM T62449 C54KPJ 11843000 IC50 = 2400 nM T62449 C63JZI 11843001 IC50 = 3800 nM T62449 CI6DR2 11843002 IC50 = 450 nM T62449 CE71YT 11843003 IC50 = 44000 nM T62449 CSW06V 11843143 IC50 > 50000 nM T62449 C0QY1S 11843144 IC50 = 620 nM T62449 CH29RF 11843145 IC50 = 970 nM T62449 CXB5U7 11843146 IC50 = 44000 nM T62449 CA2JS9 11843147 IC50 = 2200 nM T62449 CQF74N 11843148 IC50 = 2800 nM T62449 C1RB0T 11843149 IC50 = 2800 nM T62449 CRQ01W 11843150 IC50 = 340 nM T62449 CHG2O7 11843287 IC50 > 10000 nM T62449 C6AR4K 11843288 IC50 = 1300 nM T62449 C60DPL 11843289 IC50 = 21 nM T62449 C5ZF4Y 11843290 IC50 > 10000 nM T62449 C94ELW 11843291 IC50 = 5300 nM T62449 C2YV6D 11843292 IC50 > 10000 nM T62449 C9K2MI 11843293 IC50 = 4700 nM T62449 C2KVO5 11843428 IC50 = 17 nM T62449 CK1BJ7 11843429 IC50 = 26 nM T62449 C36FSN 11843430 IC50 = 310 nM T62449 C3O4LX 11843431 IC50 > 50000 nM T62449 CE5O9M 11843432 IC50 = 24000 nM T62449 CRZO78 11844343 IC50 = 300 nM T62449 C43YKI 11844344 IC50 > 10000 nM T62449 C6ET8L 11844345 IC50 = 56 nM T62449 CVNB38 11844346 IC50 = 240 nM T62449 CI3KG0 11844347 IC50 = 32 nM T62449 C0I2DQ 11844478 IC50 = 330 nM T62449 C1M3LN 11844479 IC50 > 10000 nM T62449 C1JMO5 11844480 IC50 = 74 nM T62449 CFS47B 11844481 IC50 = 4600 nM T62449 CR48MI 11844482 IC50 = 5800 nM T62449 CYUK21 11844483 IC50 = 3200 nM T62449 CWI7A5 11844484 IC50 > 10000 nM T62449 CU72HA 11844608 IC50 = 300 nM T62449 C4IM8Z 11844609 IC50 = 10000 nM T62449 CK7O0V 11844610 IC50 = 32 nM T62449 C3X5WY 11844611 IC50 = 210 nM T62449 C95MUX 11844612 IC50 = 73 nM T62449 CE50UF 11844613 IC50 = 330 nM T62449 CY2XW1 11844614 IC50 > 10000 nM T62449 CM0V7X 11844749 IC50 = 23000 nM T62449 C2A4QM 11844750 IC50 > 10000 nM T62449 CD45ER 11844751 IC50 = 260 nM T62449 CTW53J 11844752 IC50 > 10000 nM T62449 CE1L7P 11844753 IC50 > 10000 nM T62449 C51FQS 11844754 IC50 > 10000 nM T62449 C5Q1OC 11844755 IC50 = 120 nM T62449 C9JT4S 11847343 IC50 = 1634 nM T62449 C18TDF 11948705 IC50 = 8 nM T62449 C0HT7M 11951722 IC50 = 6 nM T62449 CTR9Z0 11951723 IC50 = 12 nM T62449 C4EVI9 11951724 EC50 = 12 nM T62449 CHR2C0 11951725 IC50 = 5 nM T62449 CMF5T7 11951726 IC50 = 2 nM T62449 C54TPO 11951727 IC50 = 14 nM T62449 CFYK69 11951728 IC50 = 25 nM T62449 C5M9VQ 11951901 EC50 = 8 nM T62449 C0GLF5 11952264 EC50 = 53 nM T62449 CJLB31 11952265 EC50 = 30 nM T62449 C4JE5Y 11952437 IC50 = 15 nM T62449 CS3FO8 11952438 EC50 = 40 nM T62449 CB0LK9 11952439 IC50 = 35 nM T62449 CN7VR0 11991390 IC50 = 50 nM T62449 C0EB2M 11991391 IC50 = 370 nM T62449 CPVK13 12997791 IC50 = 1080 nM T62449 CXM5P6 13000374 IC50 > 50000 nM T62449 C1AO9F 13359143 Ki = 12589.25 nM T62449 CFRS50 14809281 Ki = 31622.78 nM T62449 CY2P7U 15978890 IC50 = 49 nM T62449 C58MVQ 15978891 IC50 = 90 nM T62449 C5BFH0 15978893 IC50 = 47 nM T62449 C5XBV6 15978894 IC50 = 206 nM T62449 CCX39H 15979015 IC50 = 29 nM T62449 CRS8U6 15979020 IC50 = 60 nM T62449 CD98IU 15979137 IC50 = 29 nM T62449 CBV7T6 15979138 IC50 = 38 nM T62449 CI5Q2D 15979261 IC50 = 160 nM T62449 C2G6HB 15979262 IC50 = 120 nM T62449 C3ZC4Y 15979393 IC50 = 21 nM T62449 CSHB65 15979395 IC50 = 35 nM T62449 C6Z4CR 15979397 IC50 = 37 nM T62449 CFX2H6 15979398 IC50 = 60 nM T62449 C4D5UF 15979518 IC50 = 8 nM T62449 C1JMA7 15979519 IC50 = 6 nM T62449 CALP02 15979629 IC50 > 1050 nM T62449 CARL15 15979630 IC50 = 10 nM T62449 CM2Q8V 15979631 IC50 = 35 nM T62449 CXYU20 15979633 IC50 = 16 nM T62449 CQD02P 15979747 IC50 = 9 nM T62449 C8MGY5 15979751 IC50 = 0.03 nM T62449 CF9SK3 15979868 IC50 = 0.03 nM T62449 CFS3J0 15979870 IC50 = 0.05 nM T62449 C7UEG5 15980106 IC50 = 8 nM T62449 CPJY86 15980107 IC50 = 1.6 nM T62449 CU87FW 15980108 IC50 = 7 nM T62449 CQH37B 15980109 IC50 = 0.05 nM T62449 CT9NE3 15980231 IC50 = 1.4 nM T62449 CB7JU8 15980233 IC50 = 15 nM T62449 CA37CF 15980347 IC50 = 1 nM T62449 C7DAM4 15980349 IC50 = 0.4 nM T62449 C04XVH 15980473 IC50 = 0.05 nM T62449 CG19AY 15980475 IC50 = 12 nM T62449 C34RGF 15981966 IC50 = 400 nM T62449 CJ9T5L 15981968 IC50 = 1060 nM T62449 CNJ9H5 15982230 IC50 = 510 nM T62449 COA20K 15982231 IC50 = 12 nM T62449 CG78YR 15982234 IC50 = 17 nM T62449 C68FGK 15982236 IC50 = 440 nM T62449 C9N5YT 15982355 IC50 = 3 nM T62449 C09OAI 15982356 IC50 = 2.5 nM T62449 C1Q4HY 15982488 IC50 = 2.3 nM T62449 CF8XB2 15982612 IC50 = 2 nM T62449 CU60YX 15982613 IC50 = 0.3 nM T62449 C9NYM4 15982616 IC50 = 1.2 nM T62449 CFYB26 15982749 IC50 = 1.2 nM T62449 C5ASH4 15982884 IC50 = 25 nM T62449 CLD42C 15982885 IC50 = 11 nM T62449 C6I4CL 15982887 IC50 = 780 nM T62449 C4KF3E 15982889 IC50 = 44 nM T62449 CPW0J5 15983017 IC50 = 130 nM T62449 CFPW41 16007116 Ki > 8800 nM T62449 CB8Z1H 16040316 Ki = 12.59 nM T62449 C23TAG 16040317 EC50 = 1500 nM T62449 CLFO03 16046077 IC50 = 5100 nM T62449 CUP9C4 16046104 IC50 = 9 nM T62449 C9TU1O 16046126 IC50 > 1000 nM T62449 C2G8SU 16049816 IC50 = 1 nM T62449 CZHJ34 16058637 IC50 = 820 nM T62449 C42DYS 16091079 IC50 = 37 nM T62449 CCQ1W9 16099270 IC50 > 100000 nM T62449 CB04TO 16099272 IC50 > 100000 nM T62449 CHQL75 16099330 IC50 > 20000 nM T62449 C7VP5R 16122643 IC50 = 7 nM T62449 C8KBL7 16124892 IC50 = 11 nM T62449 C6B5LF 16124893 IC50 = 231 nM T62449 CD0V5F 16124956 IC50 = 7 nM T62449 CWC4G1 16124957 IC50 = 2 nM T62449 CSZ65C 16124958 IC50 = 4 nM T62449 CM63WR 16124959 Ki = 19.95 nM T62449 CMP31K 16124963 IC50 = 28 nM T62449 CZ9DA2 16125023 IC50 = 1 nM T62449 C7BJA9 16125024 IC50 > 10000 nM T62449 CK9ZI2 16125029 IC50 = 6 nM T62449 C45GLB 16125089 IC50 = 1060 nM T62449 CS4I8B 16125090 IC50 = 6 nM T62449 C1IY8J 16125091 IC50 = 3 nM T62449 C8JPC6 16125092 IC50 = 2 nM T62449 CL5Y7N 16125093 IC50 = 266 nM T62449 CSP25X 16125095 IC50 = 7 nM T62449 CC3SM6 16224162 IC50 = 230 nM T62449 C1HX5S 16224163 IC50 = 560 nM T62449 C1YD0E 16224363 IC50 = 1100 nM T62449 CXEL50 16224365 IC50 = 1300 nM T62449 C6DLS7 16224366 IC50 = 160 nM T62449 C4XW2Y 16224367 IC50 = 340 nM T62449 CP1KZ5 16224368 IC50 = 510 nM T62449 C5T2EM 16224369 IC50 = 17 nM T62449 CQ3W8B 16224372 IC50 = 100 nM T62449 CUWB97 16224555 IC50 = 4500 nM T62449 C5FDK3 16224560 IC50 = 18000 nM T62449 C7X8BF 16224564 IC50 = 52 nM T62449 CLFY25 16224565 IC50 = 86 nM T62449 C9FT0O 16224566 IC50 = 31 nM T62449 C8KAG5 16224568 IC50 = 100 nM T62449 C4K2CP 16224745 IC50 = 3 nM T62449 CK7HF5 16224746 IC50 = 25 nM T62449 CAZ18R 16224747 IC50 = 17 nM T62449 CL2KA1 16226178 IC50 = 130 nM T62449 CM1TO7 16226179 IC50 = 6 nM T62449 C5FHM6 16226383 IC50 = 31 nM T62449 C3ANS1 16666182 IC50 = 3 nM T62449 C1MO2D 16666228 IC50 = 14 nM T62449 CWB02U 16758227 IC50 = 1 nM T62449 CH74GF 17759184 IC50 = 893 nM T62449 C02ULI 17759310 IC50 = 43 nM T62449 CB53JQ 17759312 IC50 = 904 nM T62449 C27VPE 17759424 IC50 = 269 nM T62449 CQB4E1 17759425 IC50 = 107 nM T62449 C0DPC1 17759426 IC50 = 27 nM T62449 C46KWB 17759427 IC50 = 311 nM T62449 C4HLE3 17759428 IC50 = 161 nM T62449 C9VLS2 17759429 IC50 = 23 nM T62449 C38NQA 17759538 IC50 = 3700 nM T62449 CY1U6Q 17759539 IC50 = 1790 nM T62449 CYD7P0 18449135 Ki = 630.96 nM T62449 C1LAD6 21717212 IC50 = 4000 nM T62449 CVP75C 21914398 IC50 = 41 nM T62449 C62KMD 21980334 IC50 = 22 nM T62449 C05BIJ 21980353 IC50 = 10 nM T62449 C5H0QS 21980362 IC50 = 830 nM T62449 C13WHU 21980365 IC50 = 30 nM T62449 CQY89R 21980377 IC50 = 380 nM T62449 C39NXD 21980383 IC50 = 14 nM T62449 CX16UW 21980406 IC50 = 210 nM T62449 C75ZLY 21980427 IC50 = 134 nM T62449 CA6X4C 21980437 IC50 = 2 nM T62449 CSLM60 21980447 IC50 = 14 nM T62449 C0H5VE 21980448 IC50 = 7 nM T62449 C49MKS 21980471 IC50 = 3 nM T62449 C8V4OX 21980483 IC50 = 374 nM T62449 C6SBU7 21980490 IC50 = 730 nM T62449 CX9B0Y 21980491 IC50 = 102 nM T62449 CKBM87 21980493 IC50 = 4 nM T62449 CTP3I5 21980497 IC50 = 1700 nM T62449 C3WF0E 21980518 IC50 = 240 nM T62449 CM9DU4 21980529 IC50 = 29 nM T62449 C9C3RQ 21980545 IC50 = 5900 nM T62449 C57WSN 21980557 IC50 = 4300 nM T62449 C06IXV 21980575 IC50 = 41 nM T62449 CD7YS1 21980580 IC50 = 12 nM T62449 CTAO10 21980612 IC50 = 200 nM T62449 CQI80X 21980631 IC50 = 71 nM T62449 CP7BE6 21980647 IC50 = 22 nM T62449 CZVY24 21980658 IC50 = 36 nM T62449 C13NVO 21980695 IC50 = 290 nM T62449 CE93IF 21980705 IC50 = 770 nM T62449 CA24TJ 21980718 IC50 = 55 nM T62449 CM37OL 21980722 IC50 = 63 nM T62449 CT3QM7 21980728 IC50 = 250 nM T62449 C42ZAE 21980797 IC50 = 4700 nM T62449 C65TXJ 21980800 IC50 = 270 nM T62449 CT3YR9 21980866 IC50 = 1100 nM T62449 C7Z4LB 21980883 IC50 = 280 nM T62449 CU84GQ 21980891 IC50 = 96 nM T62449 CT6K9A 21980919 IC50 = 59 nM T62449 CD5XW2 21980923 IC50 = 74 nM T62449 CO0A5R 22064346 Ki = 6.31 nM T62449 CY0IF4 22574188 IC50 = 610 nM T62449 CJT1N5 22667253 Ki = 158.49 nM T62449 CT13RA 23627206 IC50 = 242 nM T62449 C9G5EQ 23645578 IC50 = 93000 nM T62449 C95CXB 23645579 IC50 = 21000 nM T62449 C8OZ1L 23646790 IC50 = 42 nM T62449 C6K8EC 23646791 Ki = 3.981 nM T62449 CC70LR 23646792 IC50 = 3 nM T62449 C3E8XB 23646793 IC50 = 22 nM T62449 CPSV20 23646794 IC50 = 18 nM T62449 C7OY3F 23646795 IC50 = 9 nM T62449 C8TE7B 23646796 IC50 = 15 nM T62449 CF29JX 23646797 IC50 = 23 nM T62449 CZ75ID 23646798 IC50 > 10000 nM T62449 CXA4Z8 23646799 IC50 = 11 nM T62449 CZF96K 23646800 IC50 = 9 nM T62449 CYET85 23646801 IC50 = 111 nM T62449 C2ASP4 23646802 IC50 = 42 nM T62449 CP1TD2 23646803 IC50 = 58 nM T62449 C2F9JR 23646804 IC50 = 91 nM T62449 C6VGM2 23646805 IC50 = 68 nM T62449 C7O9PI 23646806 IC50 = 243 nM T62449 CH3O6Q 23646807 IC50 = 328 nM T62449 C68NRM 23646808 IC50 = 72 nM T62449 CDI69J 23646809 IC50 = 51 nM T62449 C2XKZ4 23646810 IC50 = 1365 nM T62449 C8GZU6 23646811 IC50 = 7 nM T62449 C1G8RY 23646812 IC50 = 228 nM T62449 C3SIJ8 23646813 IC50 = 14 nM T62449 CH9QB6 23646814 IC50 = 12 nM T62449 C7QTF9 23646815 IC50 = 10 nM T62449 C48LIT 23646816 IC50 = 25 nM T62449 C50UOB 23646817 IC50 = 64 nM T62449 CGTY02 23646818 IC50 = 38 nM T62449 CU5K2W 23646820 IC50 = 66 nM T62449 CLT40P 23646821 IC50 = 38 nM T62449 CTB1M0 23646822 IC50 = 43 nM T62449 C8N4DR 23646823 IC50 = 32 nM T62449 C76IPM 23646824 IC50 = 45 nM T62449 C95SKX 23646825 IC50 = 10 nM T62449 CH90DU 23646826 IC50 = 96 nM T62449 CVIC13 23646827 IC50 = 73 nM T62449 C78MFQ 23646828 IC50 = 13 nM T62449 CN93IG 23646829 IC50 = 112 nM T62449 C0QH5J 23646830 IC50 > 50000 nM T62449 C2QAI9 23646831 IC50 = 3465 nM T62449 CW16KC 23646832 IC50 > 50000 nM T62449 CW9I5M 23646833 IC50 > 50000 nM T62449 CP5I3U 23646834 IC50 > 10000 nM T62449 CL05KG 23646835 IC50 = 29 nM T62449 CXY01F 23646836 IC50 = 1033 nM T62449 CIM78G 23646837 IC50 = 10 nM T62449 CJ3T7D 23646838 IC50 > 10000 nM T62449 CRDA69 23646839 IC50 > 10000 nM T62449 CYRF95 23646840 IC50 > 10000 nM T62449 C7DCW2 23646841 IC50 > 10000 nM T62449 C1DU3E 23646842 IC50 = 3972 nM T62449 C6KG1Q 23646843 IC50 = 25 nM T62449 C6GL4T 23646844 IC50 = 445 nM T62449 CO9KN4 23647029 IC50 = 162 nM T62449 CG6D4M 23647319 IC50 > 10000 nM T62449 CY8Z7X 23647330 IC50 > 10000 nM T62449 C4XD8H 23647348 IC50 > 10000 nM T62449 COE69L 23661658 IC50 = 2 nM T62449 CCQ64T 24180596 IC50 = 0.75 nM T62449 C1XLM5 24204009 IC50 > 100000 nM T62449 CMU75L 24204554 IC50 > 100000 nM T62449 CSM03X 24204556 IC50 > 100000 nM T62449 CB4Y6K 24204558 IC50 > 100000 nM T62449 C5GS0O 24205074 IC50 > 100000 nM T62449 CX2L1J 24755416 IC50 = 5 nM T62449 C7YG1N 24759534 IC50 = 57 nM T62449 C2UOE0 24766030 IC50 > 50000 nM T62449 CB52CV 24779778 IC50 = 72 nM T62449 CJF74R 24779781 IC50 = 92 nM T62449 C9E1AT 24779782 IC50 = 190 nM T62449 C0MO8J 24800837 IC50 > 100000 nM T62449 C50PMF 24813538 IC50 > 5000 nM T62449 C1LB6F 24813540 IC50 = 210 nM T62449 CT2BX4 24815996 IC50 = 87 nM T62449 CLM4R6 24815997 IC50 = 390 nM T62449 CA48TY 24815998 IC50 = 610 nM T62449 CCP2M3 24822704 IC50 > 50000 nM T62449 CUBO36 24824518 IC50 = 28 nM T62449 CNT26R 24824678 IC50 = 34000 nM T62449 C4ST1C 24824679 IC50 = 2200 nM T62449 C8FO4R 24824680 IC50 = 21 nM T62449 CI5B6S 24825779 IC50 > 50000 nM T62449 CP5EL9 24884696 IC50 = 170 nM T62449 CTFS94 24884697 IC50 = 200 nM T62449 C70ZFW 24884912 IC50 = 54 nM T62449 C0WG1I 24884913 IC50 = 360 nM T62449 CJ1SQ0 24884914 IC50 = 27 nM T62449 C98IDB 24884915 IC50 > 10000 nM T62449 CQ3S5Y 24884916 IC50 = 54 nM T62449 CGN52J 24884917 IC50 = 110 nM T62449 C0OJM4 24885126 IC50 = 850 nM T62449 C68PXG 24885315 IC50 = 3400 nM T62449 CWAL41 24885316 IC50 = 21 nM T62449 CY8L7E 24896769 IC50 > 10000 nM T62449 CNJ89Y 24939280 IC50 = 24 nM T62449 CLZ23U 24951610 EC50 = 30 nM T62449 CKP8Q1 24952336 EC50 = 100 nM T62449 C4KT5N 24954092 IC50 = 4 nM T62449 C6WZA1 24955889 IC50 = 38 nM T62449 CG5W8U 24955890 IC50 = 280 nM T62449 CW07NP 24956254 IC50 = 1300 nM T62449 C57OCS 24956256 IC50 = 8 nM T62449 CVI05A 24956257 IC50 = 4000 nM T62449 CC86JT 24956259 IC50 = 39 nM T62449 CXCU10 24956609 IC50 = 38 nM T62449 C9A1TI 24956966 IC50 = 110 nM T62449 C65LGP 24956971 IC50 = 5700 nM T62449 C5BW7I 24967393 IC50 = 240 nM T62449 C3IMA7 24967756 IC50 = 11000 nM T62449 CV9I5X 24968112 IC50 > 50000 nM T62449 CDJ17S 24968115 IC50 = 6900 nM T62449 CM8S5J 24968116 IC50 = 4500 nM T62449 CDZ72E 24968117 EC50 = 3750 nM T62449 CGL5K1 24968460 EC50 = 40 nM T62449 CE1XL0 24968463 IC50 = 2 nM T62449 CN3O5D 24968464 EC50 = 7500 nM T62449 C4EG8R 24993189 IC50 > 10000 nM T62449 CBK82P 25011729 IC50 > 30000 nM T62449 CX1HL8 25032704 Ki > 8780 nM T62449 C05OZY 25068614 IC50 = 430 nM T62449 C49SOH 25068616 IC50 = 3200 nM T62449 C2KY1G 25094210 IC50 = 187 nM T62449 CMBU37 25094945 IC50 = 87 nM T62449 CIE52F 25095213 IC50 = 19 nM T62449 C90VFX 25095214 IC50 = 36 nM T62449 CQX01F 25095215 EC50 = 10000 nM T62449 C49UDB 25095216 EC50 = 2500 nM T62449 CS1D3K 25095480 IC50 = 7 nM T62449 C8JRS1 25095481 IC50 = 19 nM T62449 CJ32BM 25095482 IC50 = 69 nM T62449 C2Z3HE 25095483 IC50 = 5 nM T62449 C6R8BY 25095485 EC50 = 3500 nM T62449 CBU47I 25095741 IC50 = 89 nM T62449 CW45BY 25095743 IC50 = 55 nM T62449 CL65JN 25095744 IC50 = 120 nM T62449 COM47Y 25095999 IC50 = 86 nM T62449 CBM20C 25096000 EC50 = 1000 nM T62449 C6C2EZ 25096003 EC50 = 1250 nM T62449 C8PR9O 25096004 IC50 = 28 nM T62449 CV2DG6 25096256 IC50 = 430 nM T62449 CGT1W6 25144294 IC50 = 20 nM T62449 CU7VR0 25144732 IC50 = 13 nM T62449 C6BWZ8 25145145 IC50 = 640 nM T62449 C78YWA 25145716 IC50 = 360 nM T62449 C6FGQ1 25206346 IC50 > 10000 nM T62449 CNG96H 25210579 IC50 > 10000 nM T62449 CH7OJ6 25221980 IC50 = 1700 nM T62449 CQKH23 25222088 IC50 = 1700 nM T62449 C6SO9B 25222091 IC50 = 670 nM T62449 CI9P4F 25222092 IC50 = 290 nM T62449 C75FIT 25222313 IC50 = 3700 nM T62449 CW58XI 25222318 IC50 = 2300 nM T62449 CB9KL2 25222319 IC50 = 3000 nM T62449 COPW43 42610049 IC50 = 22000 nM T62449 CPBZ35 42610232 IC50 = 21 nM T62449 CTCM25 42610483 IC50 = 130 nM T62449 C3Q4ZI 42610562 IC50 = 1500 nM T62449 C6NY2D 42610563 IC50 = 2500 nM T62449 CBQ1W8 42610564 IC50 = 400 nM T62449 CAZ13J 42610708 IC50 = 20000 nM T62449 C8UB2R 42610777 IC50 = 1800 nM T62449 C5C3LW 44120114 Ki = 7.943 nM T62449 CZK64Q 44129608 IC50 = 860 nM T62449 C92QHS 44133237 IC50 = 3 nM T62449 CU8P3N 44133238 IC50 = 5 nM T62449 CLW80F 44160269 IC50 = 4500 nM T62449 CO6HU7 44178069 IC50 = 100 nM T62449 CQ3OK0 44182389 IC50 = 51 nM T62449 C9P3IB 44184073 IC50 = 0.3 nM T62449 CA52KO 44184233 IC50 = 20.8 nM T62449 CSIH59 44184234 IC50 = 12 nM T62449 C1DY6A 44184236 IC50 = 0.4 nM T62449 CM0FQ6 44184237 IC50 = 0.6 nM T62449 CIEG48 44184394 IC50 = 0.5 nM T62449 CC6SR5 44184395 IC50 = 0.4 nM T62449 CCI50O 44184540 IC50 = 12.8 nM T62449 C7IE2N 44184686 IC50 = 15.1 nM T62449 C16LJD 44189155 IC50 = 290 nM T62449 CK2C6M 44193487 IC50 = 21000 nM T62449 CI7YG4 44193488 IC50 = 2800 nM T62449 COU85V 44203745 IC50 = 22 nM T62449 C3XP0I 44203747 IC50 = 3.8 nM T62449 C7R1QT 44203849 IC50 = 27 nM T62449 CT08EG 44203851 IC50 = 560 nM T62449 C0FPD7 44203853 IC50 = 7 nM T62449 CL3UT1 44203854 IC50 = 23 nM T62449 CJ7AF4 44203948 IC50 = 6.1 nM T62449 CFZT40 44203954 IC50 = 49 nM T62449 CB1TL0 44204444 IC50 = 1900 nM T62449 C57QDT 44204448 IC50 = 9000 nM T62449 CU7R0F 44205165 IC50 = 940 nM T62449 CG1VH9 44205166 IC50 = 17 nM T62449 CHQ7R3 44205167 IC50 = 740 nM T62449 CK73NR 44219749 IC50 > 50000 nM T62449 C8PQA1 44220913 IC50 = 9200 nM T62449 CW4GS7 44221131 IC50 = 390 nM T62449 C2QW3C 44221132 IC50 = 890 nM T62449 C4B5HM 44221133 IC50 = 700 nM T62449 CG3W4C 44224009 Ki = 146 nM T62449 CH94TA 44246252 IC50 = 1000 nM T62449 CWQ5F1 44410360 IC50 = 15 nM T62449 CV09DY 44410717 IC50 > 10000 nM T62449 CP3CI1 44410720 IC50 > 10000 nM T62449 C8W7AD 44410723 IC50 > 10000 nM T62449 CAT5X4 44410829 IC50 > 10000 nM T62449 CC6Y5P 44410844 IC50 > 10000 nM T62449 CG34TY 44410851 IC50 > 10000 nM T62449 C41EIA 44410869 IC50 > 10000 nM T62449 CB6AE8 44410948 IC50 > 10000 nM T62449 CXZG12 44410949 IC50 > 10000 nM T62449 CS7IE9 44410953 IC50 > 10000 nM T62449 CA9M4X 44410954 IC50 > 10000 nM T62449 C3SP5H 44410955 IC50 > 10000 nM T62449 C5D6YP 44410956 IC50 > 10000 nM T62449 C5W1VC 44410959 IC50 > 10000 nM T62449 CM1C2G 44410960 IC50 > 10000 nM T62449 CVSI80 44411048 IC50 > 10000 nM T62449 CN72BR 44411161 IC50 > 10000 nM T62449 C4AW0O 44411183 IC50 > 10000 nM T62449 C6H9GQ 44415009 IC50 = 10000 nM T62449 CAHI52 44419928 IC50 = 4 nM T62449 C98IAF 44419929 EC50 = 3900 nM T62449 CM1HR8 44419935 EC50 = 170 nM T62449 COJM58 44419936 EC50 = 460 nM T62449 C9VK6T 44419941 EC50 = 520 nM T62449 CC5F1P 44419945 IC50 = 5.6 nM T62449 C5ZA6O 44419946 IC50 = 4.3 nM T62449 CF48CY 44419952 EC50 = 130 nM T62449 C92ZIB 44419957 EC50 = 190 nM T62449 C9JSN2 44419975 IC50 = 29 nM T62449 C94PLN 44419976 IC50 = 20 nM T62449 CQN2G9 44419980 IC50 = 0.83 nM T62449 CEDA70 44419982 EC50 = 420 nM T62449 CCV9H1 44419986 EC50 = 870 nM T62449 C7R9FY 44419987 IC50 = 2.1 nM T62449 C3E5RU 44420002 IC50 = 580 nM T62449 CBWG73 44420003 IC50 = 190 nM T62449 CN9D1X 44427496 IC50 > 10000 nM T62449 CA3H1N 44427497 IC50 = 3600 nM T62449 CPG36L 44427498 IC50 = 500 nM T62449 CC3M9Q 44427499 IC50 > 10000 nM T62449 COHK14 44427500 IC50 > 10000 nM T62449 CM05CR 44427501 IC50 = 8000 nM T62449 COBM60 44427502 IC50 = 2100 nM T62449 C7WC5Z 44427503 IC50 > 10000 nM T62449 C10NBU 44427504 IC50 > 10000 nM T62449 C3TI0U 44427505 IC50 > 10000 nM T62449 C1SP6M 44427506 IC50 = 72 nM T62449 CKB9U7 44427507 IC50 = 11 nM T62449 C84VCD 44427508 IC50 = 14 nM T62449 CJ5Y4B 44427509 IC50 = 16 nM T62449 C0ES3O 44427510 IC50 = 104 nM T62449 CE0VO8 44427511 IC50 = 17 nM T62449 C3E7RV 44427512 IC50 = 2 nM T62449 C2QIV3 44427513 IC50 = 4 nM T62449 CGJZ06 44427514 IC50 = 6 nM T62449 CN1YZ8 44427515 EC50 = 2100 nM T62449 CU6VP1 44427516 EC50 = 890 nM T62449 C7WDA1 44427517 EC50 = 2630 nM T62449 CETQ79 44427518 IC50 = 7 nM T62449 COPG94 44427519 IC50 = 6.7 nM T62449 CU7NW8 44427520 IC50 = 2 nM T62449 C7YTE1 44427521 IC50 = 10 nM T62449 CR9WL8 44427522 IC50 = 6 nM T62449 CHSK01 44427523 IC50 = 10 nM T62449 CXE02T 44427524 IC50 = 1640 nM T62449 C0W8VE 44427525 IC50 = 910 nM T62449 CSN17U 44428979 IC50 = 459 nM T62449 C7SPC8 44428980 IC50 = 1473 nM T62449 C9D2LT 44428981 IC50 = 481 nM T62449 CPG3Y1 44428982 IC50 = 1042 nM T62449 CLD2H1 44428983 IC50 = 497 nM T62449 CNW25X 44428984 IC50 = 790 nM T62449 CSV2N1 44428985 IC50 = 966 nM T62449 CJX2L1 44428986 IC50 = 1600 nM T62449 CKC3W0 44428987 IC50 = 2044 nM T62449 CGM64V 44428988 IC50 = 5260 nM T62449 CE5KB7 44428989 IC50 = 602 nM T62449 CX1G7J 44428993 IC50 = 12 nM T62449 C79GOK 44428995 IC50 = 535 nM T62449 CQSE96 44428996 IC50 = 8742 nM T62449 CMK9I6 44428997 IC50 = 4825 nM T62449 CX07ZP 44428999 IC50 = 1029 nM T62449 C67HSD 44429000 IC50 = 3064 nM T62449 CT0S9B 44429001 IC50 = 1880 nM T62449 CRV73D 44429002 IC50 = 6472 nM T62449 C9W6PN 44434777 IC50 > 10000 nM T62449 CV4S1N 44434779 IC50 = 15 nM T62449 CRQL06 44434783 IC50 = 5 nM T62449 CQT20Z 44434784 IC50 = 6 nM T62449 CE34MW 44434786 IC50 = 5 nM T62449 CSPE59 44434791 IC50 = 16 nM T62449 C4FV5L 44434798 IC50 = 12 nM T62449 C9B7HF 44434800 IC50 = 108 nM T62449 CCN3J2 44434823 IC50 = 25 nM T62449 CM68VT 44434827 IC50 = 55 nM T62449 CI5YT2 44434832 IC50 = 7 nM T62449 CXCF61 44434837 IC50 = 3 nM T62449 CRF16E 44434842 IC50 = 3 nM T62449 CVD15Z 44434844 IC50 = 8 nM T62449 CVF0D7 44434846 IC50 = 16 nM T62449 C5CYI7 44434852 IC50 = 11 nM T62449 C4QWM0 44434866 IC50 = 4 nM T62449 CNI43Z 44434869 IC50 = 4 nM T62449 CWD65M 44434871 IC50 = 2 nM T62449 CXSD73 44434873 IC50 = 2 nM T62449 C3VF1Q 44434874 IC50 = 4 nM T62449 C2NJ3T 44434875 IC50 = 3 nM T62449 C9PY7H 44434957 IC50 = 31 nM T62449 C3MC1S 44434961 IC50 = 22 nM T62449 C5GDS4 44442329 IC50 = 0.8 nM T62449 C3I5CJ 44442336 IC50 = 3.7 nM T62449 C2T7YV 44442339 IC50 = 3.8 nM T62449 C7BJ1C 44442340 IC50 = 2.5 nM T62449 CY1X9O 44442341 IC50 = 3.1 nM T62449 CTJ56F 44442342 IC50 = 3 nM T62449 CHQ1N7 44442343 IC50 = 1.1 nM T62449 C34KOH 44442344 IC50 = 2.6 nM T62449 CSW9Z7 44442345 IC50 = 52 nM T62449 CC8IS6 44442346 IC50 = 6.4 nM T62449 CU9M8W 44442347 IC50 = 5.9 nM T62449 CVXH13 44442348 IC50 = 1.8 nM T62449 C86NJL 44442349 IC50 = 1 nM T62449 CKY4J3 44442350 IC50 = 1.5 nM T62449 CH6I5T 44442353 IC50 = 1.1 nM T62449 C28FTX 44442355 IC50 = 1.5 nM T62449 C1NW0D 44442358 IC50 = 0.92 nM T62449 CZA7N5 44442360 IC50 = 2.6 nM T62449 CSF4D6 44442361 IC50 = 1 nM T62449 CRLA52 44442362 IC50 = 3.2 nM T62449 C1UAB7 44442363 IC50 = 1.4 nM T62449 CC3A2W 44442364 IC50 = 7 nM T62449 CN38SI 44442365 IC50 = 16 nM T62449 CK82OM 44442366 IC50 = 1.2 nM T62449 CY3ZH7 44442367 IC50 = 6.5 nM T62449 CL43MK 44442368 IC50 = 6.4 nM T62449 CAI51R 44443117 IC50 = 7 nM T62449 C4PI3E 44443121 IC50 = 2 nM T62449 CEIB19 44443123 IC50 = 25 nM T62449 CNW65X 44443126 IC50 = 779 nM T62449 CSHM05 44443128 IC50 = 355 nM T62449 CKX2M0 44443133 IC50 > 10000 nM T62449 CR1J4S 44443134 IC50 = 73 nM T62449 CS1H7Q 44443135 IC50 > 10000 nM T62449 CL14DT 44443163 IC50 = 1288 nM T62449 C0VMC7 44443164 IC50 = 6223 nM T62449 CI63DR 44443165 IC50 = 4579 nM T62449 CNM85X 44443166 IC50 = 11 nM T62449 CYQ73R 44443167 IC50 = 47 nM T62449 CQ7ZV5 44443168 IC50 = 77 nM T62449 CQ5GT6 44443169 IC50 = 1260 nM T62449 CNYZ27 44443170 IC50 = 1374 nM T62449 CQC29Z 44443171 IC50 = 3709 nM T62449 CTK63P 44443172 IC50 = 3003 nM T62449 CJ83RS 44443173 IC50 = 5140 nM T62449 COB1N4 44443174 IC50 = 19 nM T62449 CGAY03 44443175 IC50 = 5 nM T62449 CH47GW 44443176 IC50 > 10000 nM T62449 CL1F7I 44443177 IC50 = 1743 nM T62449 C4JK5E 44443178 IC50 > 10000 nM T62449 CF5G0A 44443180 IC50 = 15 nM T62449 CI0CW5 44443181 IC50 = 4 nM T62449 CF9UN0 44443182 IC50 = 2 nM T62449 C1PH2S 44443183 IC50 = 288 nM T62449 CGWT05 44443184 IC50 = 288 nM T62449 C7R6IO 44443185 IC50 = 16 nM T62449 C1UKD9 44443186 IC50 > 10000 nM T62449 CDV09P 44443187 IC50 = 44 nM T62449 C6S5HU 44443188 IC50 = 89 nM T62449 CV4EJ5 44443189 IC50 = 44 nM T62449 CFJ9B7 44443190 IC50 = 4 nM T62449 CMR7L3 44443191 IC50 = 3 nM T62449 CN63XD 44443192 IC50 = 3 nM T62449 CO2LA0 44443193 IC50 = 6 nM T62449 CIP70H 44443196 IC50 = 14 nM T62449 C2MSQ4 44443197 IC50 = 20 nM T62449 C9XWJ6 44443205 IC50 = 10 nM T62449 CQ15OX 44443207 IC50 = 77 nM T62449 C2S6XE 44443209 IC50 = 9 nM T62449 CT3UM2 44443212 IC50 = 3 nM T62449 C3LCB2 44443215 IC50 = 2 nM T62449 C2VZE5 44443217 IC50 = 1 nM T62449 C1N4YK 44443220 IC50 = 3 nM T62449 C7UES0 44443223 IC50 = 17 nM T62449 CWF5I3 44443283 IC50 = 6 nM T62449 C0GI4W 44443507 IC50 = 360 nM T62449 CU5V4G 44443509 IC50 = 300 nM T62449 C3SM6F 44443512 IC50 = 420 nM T62449 C6G4FY 44443515 IC50 = 11 nM T62449 CZ0N9F 44443518 IC50 = 3 nM T62449 CG30PL 44443519 IC50 = 3.5 nM T62449 CXW58E 44443521 IC50 = 4.3 nM T62449 CISV72 44443522 IC50 = 0.5 nM T62449 C8R1XO 44443523 IC50 = 2.4 nM T62449 CNB5A4 44443524 IC50 = 9.2 nM T62449 CZ2UK4 44443525 IC50 = 6.5 nM T62449 C2O5EX 44443526 IC50 = 0.6 nM T62449 C2LSP8 44443527 IC50 = 2 nM T62449 C3LF7I 44443536 IC50 = 3.6 nM T62449 C7HUA2 44443537 IC50 = 2 nM T62449 CXF3E8 44443539 IC50 = 2.6 nM T62449 C1PY0A 44443542 IC50 = 3.7 nM T62449 CRH5N2 44443544 IC50 = 3.5 nM T62449 C30SRZ 44443546 IC50 = 0.8 nM T62449 CB2GO3 44443549 IC50 = 11.5 nM T62449 CNEO01 44443782 IC50 = 18 nM T62449 C0MCW6 44443784 IC50 = 12 nM T62449 CK9R3S 44443786 IC50 = 10 nM T62449 CA9K6M 44443788 IC50 = 850 nM T62449 C0Z2QN 44443789 IC50 = 64 nM T62449 C7QU9M 44443790 IC50 = 60 nM T62449 CBT41I 44443791 IC50 = 220 nM T62449 C9IS0N 44443794 IC50 = 36 nM T62449 CI2T9K 44443797 IC50 = 20 nM T62449 CXQP15 44443798 IC50 = 1.1 nM T62449 CV8Y2S 44443800 IC50 = 14 nM T62449 C41ECU 44443802 IC50 = 3.2 nM T62449 CUHO63 44443803 IC50 = 3.1 nM T62449 CT08MR 44444773 IC50 = 0.3 nM T62449 C3K6XO 44444776 IC50 = 2 nM T62449 CD4JN8 44444778 IC50 = 2 nM T62449 CG9F5Z 44444779 IC50 = 1 nM T62449 CJI0V3 44444780 IC50 = 2 nM T62449 C0SH3K 44444781 IC50 = 4 nM T62449 C29YMW 44444782 IC50 = 6 nM T62449 C5H7EK 44444783 IC50 = 6 nM T62449 CV6S1E 44444784 IC50 = 3 nM T62449 CJQ06A 44444814 IC50 = 3 nM T62449 CZT5C8 44444827 IC50 = 10 nM T62449 C25MTH 44444831 IC50 = 1 nM T62449 C13BEO 44444834 IC50 = 2 nM T62449 CI34PG 44444835 IC50 = 1 nM T62449 C5N4WV 44444836 IC50 = 0.3 nM T62449 CFI34Q 44444837 IC50 = 1 nM T62449 C42NLA 44444838 IC50 = 1 nM T62449 CWS13R 44444839 IC50 = 2 nM T62449 CB4C8D 44444840 IC50 = 2 nM T62449 C2OX0Q 44444841 IC50 = 23 nM T62449 CO9AZ3 44444842 IC50 = 3 nM T62449 CTVP72 44444844 IC50 = 4 nM T62449 C3K4HX 44444845 IC50 = 4 nM T62449 CGB39X 44444846 IC50 = 3 nM T62449 CA8JQ9 44444847 IC50 = 6 nM T62449 C9MO1U 44444849 IC50 = 8 nM T62449 CLV5E4 44444850 IC50 = 8 nM T62449 C4Z9VK 44444851 IC50 = 1 nM T62449 C3AJG6 44444852 IC50 = 3 nM T62449 C5S8JM 44444853 IC50 = 1 nM T62449 CDAF04 44444854 IC50 = 1 nM T62449 C3HX8P 44452464 IC50 = 1920 nM T62449 C3LYA8 44452483 IC50 = 14500 nM T62449 CA09HX 44453136 IC50 = 0.98 nM T62449 C93EWR 44453137 EC50 = 3100 nM T62449 CH91LC 44453138 EC50 = 2000 nM T62449 C17IZO 44453174 EC50 = 3100 nM T62449 C2Z4CX 44453205 EC50 = 280 nM T62449 CPR1Q9 44453209 EC50 = 70 nM T62449 CV01FK 44453299 EC50 = 220 nM T62449 CUAV84 44453331 EC50 = 350 nM T62449 C96YMZ 44453333 EC50 = 3500 nM T62449 C5IZV3 44453371 IC50 = 11.2 nM T62449 C4GRV3 44453411 IC50 = 3.5 nM T62449 C7FTE1 44453478 EC50 = 40 nM T62449 C67XRE 44453479 IC50 = 7.9 nM T62449 CET02I 44453508 IC50 = 22 nM T62449 C3GH1E 44453537 EC50 = 600 nM T62449 CT8MI5 44453564 EC50 = 2100 nM T62449 CMU3B7 44453590 IC50 = 8.1 nM T62449 C4A8IN 44453591 IC50 = 4.8 nM T62449 CK8GA9 44453622 EC50 = 50 nM T62449 C8AG7J 44453623 IC50 = 4 nM T62449 CR1E5P 44453624 IC50 = 1050 nM T62449 CRJ8F6 44454116 IC50 = 44 nM T62449 CWZ0L4 44454457 IC50 = 57 nM T62449 CYH6P3 44520205 IC50 > 10000 nM T62449 C8LJS5 44520782 IC50 = 1100 nM T62449 CNI56K 44520783 IC50 = 8500 nM T62449 CN4R3E 44520784 IC50 = 5200 nM T62449 CN5V6I 44520785 IC50 = 2500 nM T62449 CJ1K0O 44525558 IC50 = 2300 nM T62449 C5L8AQ 44545550 IC50 = 1.1 nM T62449 C02WLM 44545753 EC50 = 168 nM T62449 CXY10R 44545757 IC50 = 1 nM T62449 COY01J 44545824 EC50 = 216 nM T62449 C86IVN 44545828 EC50 = 99.1 nM T62449 CI0VW1 44545897 IC50 = 78.7 nM T62449 CRWT79 44545901 IC50 = 1.3 nM T62449 C96YPZ 44546167 IC50 = 0.78 nM T62449 CS5OI0 44546169 EC50 = 658 nM T62449 CT30BJ 44546231 IC50 = 41.7 nM T62449 CZH21K 44546426 IC50 = 1.3 nM T62449 CATK49 44546490 EC50 = 656 nM T62449 COZ20N 44546493 IC50 = 0.95 nM T62449 CLJ98C 44560372 IC50 < 10 nM T62449 C32EOZ 44560373 IC50 = 7 nM T62449 C7QFG5 44560374 IC50 = 9 nM T62449 C8I5MG 44560375 IC50 = 11 nM T62449 CMK86D 44560523 IC50 = 5 nM T62449 C3JLV0 44560524 IC50 = 10 nM T62449 CD0G2Q 44560525 IC50 = 6 nM T62449 C6N8KF 44560526 IC50 = 19 nM T62449 CR5J0U 44560570 IC50 = 13 nM T62449 CJ10TV 44560571 IC50 = 41 nM T62449 CU5BJ6 44560572 IC50 = 8 nM T62449 C2T5SV 44560573 IC50 = 41 nM T62449 CFH04Q 44560574 IC50 = 6 nM T62449 CF8YC0 44560617 IC50 = 7 nM T62449 CZ01JT 44560618 IC50 = 3 nM T62449 CW35LK 44560619 IC50 = 6 nM T62449 CLUR57 44560620 IC50 = 6 nM T62449 CGP4W3 44560621 IC50 = 4 nM T62449 CBTA02 44560667 IC50 = 5 nM T62449 CX2HY8 44560668 IC50 = 9 nM T62449 CT2WY9 44560669 IC50 = 9 nM T62449 CE6P3S 44560670 IC50 = 10 nM T62449 C9MS1V 44560703 IC50 > 30000 nM T62449 C4U9NW 44560704 IC50 = 110 nM T62449 CF03RB 44560705 IC50 = 170 nM T62449 CRGF45 44560706 IC50 = 160 nM T62449 C0IUL2 44560707 IC50 = 600 nM T62449 C2P9SF 44560752 IC50 > 300 nM T62449 CRN67T 44560753 IC50 = 360 nM T62449 CQK8Z9 44560771 IC50 = 230 nM T62449 CZQ5D1 44560772 IC50 = 6700 nM T62449 CWR6V4 44560805 IC50 = 2600 nM T62449 CR6XC0 44560806 IC50 = 31 nM T62449 CKV64F 44560807 IC50 = 39 nM T62449 CCAB70 44560808 IC50 = 29 nM T62449 CJ6W3X 44560831 IC50 = 17 nM T62449 C2L6XP 44560879 IC50 > 10000 nM T62449 CRAJ61 44560880 IC50 = 2100 nM T62449 CC46NO 44560909 IC50 = 3900 nM T62449 C1CP0U 44560910 IC50 = 5100 nM T62449 C0KBL9 44560911 IC50 = 7100 nM T62449 CS7WA4 44560912 IC50 = 30 nM T62449 CA7TR0 44560913 IC50 = 100 nM T62449 C6Y0BC 44560914 IC50 = 110 nM T62449 CA54KS 44560935 IC50 = 5500 nM T62449 C1W7BE 44560936 IC50 = 100 nM T62449 CZHW38 44560937 IC50 = 100 nM T62449 CDR2E6 44560938 IC50 = 300 nM T62449 CG0F8K 44560939 IC50 = 3 nM T62449 CYAZ26 44560971 IC50 = 23000 nM T62449 C1ICG7 44560972 IC50 = 110 nM T62449 C87DHK 44560973 IC50 = 130 nM T62449 C3ZPH8 44560974 IC50 = 980 nM T62449 C30LTJ 44576328 IC50 = 5000 nM T62449 CK4S7Z 44576333 IC50 = 5000 nM T62449 CD3SR9 44576334 IC50 = 1320 nM T62449 CKR05I 44576335 IC50 = 25 nM T62449 C3T1HQ 44576337 IC50 = 14 nM T62449 C2BGJ1 44576358 IC50 = 27 nM T62449 CZUH48 44591031 IC50 > 100000 nM T62449 CC5LK9 44591032 IC50 > 100000 nM T62449 C8E0LW 44591039 IC50 = 20000 nM T62449 CW62ZA 44591040 IC50 = 21000 nM T62449 CU69LX 44591041 IC50 = 1300 nM T62449 CH35PV 44591070 IC50 = 17000 nM T62449 C5PM9O 44591072 IC50 > 100000 nM T62449 CWI2X6 44591073 IC50 = 3300 nM T62449 CG60AL 44591074 IC50 = 6000 nM T62449 CAXI82 44591075 IC50 = 3800 nM T62449 CIUO70 44591076 IC50 = 4500 nM T62449 C0LX3R 44591077 IC50 > 100000 nM T62449 CFRY37 44591080 IC50 = 41000 nM T62449 C16HDQ 44591081 IC50 > 100000 nM T62449 C5RPU7 44591082 IC50 > 100000 nM T62449 C4YCX6 44591084 IC50 = 28000 nM T62449 CZH7A9 44591085 IC50 = 17000 nM T62449 C7H6TB 44594105 IC50 = 675 nM T62449 C28QLM 44605035 IC50 > 50000 nM T62449 C75XHS 44605037 IC50 > 50000 nM T62449 CU3RF1 45139989 IC50 > 10000 nM T62449 CQGZ06 45139991 IC50 > 10000 nM T62449 C7NQ5X 45266934 Ki = 398.11 nM T62449 CNS94R 45266971 Ki = 19.95 nM T62449 C09CVH 45266972 Ki = 2.512 nM T62449 CNJB06 45267005 Ki = 1.259 nM T62449 CVG5L0 45267033 Ki = 1.995 nM T62449 C9B3QM 45267785 Ki = 6.31 nM T62449 C1TIB6 45267786 Ki = 5.012 nM T62449 CJ37RP 45267789 Ki = 63.1 nM T62449 C9GX6O 45267794 Ki = 1258.93 nM T62449 CL3H6C 45267801 Ki = 398.11 nM T62449 CA59GX 45268672 Ki = 10 nM T62449 CSER04 45268673 Ki = 10 nM T62449 CP5K0C 45268685 Ki = 125.89 nM T62449 C3RMC1 45268686 Ki = 398.11 nM T62449 C09RZC 45268690 Ki = 6309.57 nM T62449 CD0LU8 45269528 Ki = 2.512 nM T62449 CG5ZD2 45269532 Ki = 1000 nM T62449 CFW36D 45269533 Ki = 2.512 nM T62449 CPFT90 45269535 Ki = 3981.07 nM T62449 C7BTM0 45269536 Ki = 125.89 nM T62449 CRQN46 45269538 Ki = 2511.89 nM T62449 CSR84B 45269543 Ki = 39.81 nM T62449 C1U8JK 45269548 Ki = 100 nM T62449 C4H5NV 45269552 Ki = 794.33 nM T62449 C2KRI8 45269554 Ki = 125.89 nM T62449 CZ8B2L 45270354 Ki = 3.162 nM T62449 C19UND 45270355 Ki = 15.85 nM T62449 CO59EJ 45270356 Ki = 5.012 nM T62449 C0VJA9 45270357 Ki = 199.53 nM T62449 CNDA15 45270361 Ki = 10 nM T62449 C2DMA6 45270362 Ki = 15.85 nM T62449 C6RJ5G 45270363 Ki = 39.81 nM T62449 CH95GC 45270364 Ki = 0.631 nM T62449 CEW71Z 45270365 Ki = 251.19 nM T62449 C8X1HW 45270366 Ki = 5.012 nM T62449 CVZ0F5 45271175 Ki = 12.59 nM T62449 CG78NM 45271177 Ki = 10 nM T62449 CRP85E 45271179 Ki = 79.43 nM T62449 C07DTO 45271183 Ki = 79.43 nM T62449 C2OC9U 45271186 Ki = 1.585 nM T62449 C8S1PU 45272083 Ki = 12.59 nM T62449 C9AWL7 45272085 Ki = 125.89 nM T62449 C8KB6J 45272086 Ki = 31.62 nM T62449 C7ZQ1F 45272087 Ki = 39810.72 nM T62449 C14RKH 45272088 Ki = 3.981 nM T62449 C4XU7W 45272092 Ki = 15.85 nM T62449 CL3R5A 45272915 Ki = 1.585 nM T62449 CYOB37 45272920 Ki = 25.12 nM T62449 CUH91F 45272921 Ki = 251.19 nM T62449 CA5F8D 45272926 Ki = 3162.28 nM T62449 CNI82F 45272928 Ki = 50.12 nM T62449 C96LYJ 45272935 Ki = 5.012 nM T62449 CC95PQ 45375865 IC50 > 50000 nM T62449 CEOQ27 45375866 IC50 > 50000 nM T62449 C6E2SC 45482700 IC50 > 10000 nM T62449 CZXH74 45482750 IC50 > 10000 nM T62449 CUA97D 46209401 IC50 = 1400 nM T62449 CZY9T4 46212930 IC50 = 22 nM T62449 CQX0E9 46213698 IC50 = 448 nM T62449 C5L3RW 46213764 IC50 = 336 nM T62449 C7O2ND 46213766 IC50 = 251 nM T62449 C84LBR 46213822 IC50 = 123 nM T62449 CSVU49 46213824 IC50 = 235 nM T62449 C93YQM 46213881 IC50 = 31 nM T62449 C41ASQ 46213883 IC50 = 46 nM T62449 C8QG1H 46213885 IC50 = 2.8 nM T62449 CZ58FY 46215814 IC50 > 10000 nM T62449 CY3HW5 46224684 IC50 = 2800 nM T62449 CJ9W4F 46229795 IC50 = 3000 nM T62449 CHE6Z4 46229985 IC50 = 4000 nM T62449 C09ANB 46229988 IC50 = 2000 nM T62449 CT82YZ 46230040 IC50 = 3500 nM T62449 CGZT61 46230090 IC50 = 8900 nM T62449 CV5UG7 46230182 IC50 = 3400 nM T62449 C2C0MI 46230184 IC50 = 780 nM T62449 CGNX36 46230185 IC50 = 2500 nM T62449 C7ON5A 46233287 IC50 > 10000 nM T62449 CT1E0W 46238916 IC50 = 3 nM T62449 COTJ39 46863083 IC50 = 310 nM T62449 C0F9RH 46863195 IC50 = 27 nM T62449 C5FMC8 46863199 IC50 = 690 nM T62449 CLD1W7 46863317 IC50 = 290 nM T62449 C64LIW 46863435 IC50 = 890 nM T62449 C0CXG9 46863436 IC50 = 5070 nM T62449 CA4QB7 46863552 IC50 = 23 nM T62449 CO3P0J 46866604 IC50 < 50000 nM T62449 CLS29B 46872626 IC50 > 10000 nM T62449 CJOM49 46880136 IC50 = 18600 nM T62449 C2O8RZ 46886323 IC50 > 1000 nM T62449 CWM49L 46911672 IC50 = 199526231.5 nM T62449 CDX8G4 46911673 IC50 = 660693448 nM T62449 CRXG74 46911674 IC50 = 501187233.6 nM T62449 CZ3XP5 46926535 IC50 > 100000 nM T62449 C1G5ND 46932941 IC50 = 0.5 nM T62449 C5NBQ3 46932942 IC50 = 1 nM T62449 CF2PN5 46933087 IC50 = 0.6 nM T62449 CBR6M2 46934729 IC50 = 0.1 nM T62449 C5GOV0 46934730 IC50 = 4 nM T62449 C91UDR 49786973 IC50 = 1 nM T62449 CSKM74 49797811 IC50 = 28000 nM T62449 CDB5V3 49797812 IC50 = 3500 nM T62449 CNI52G 49797813 IC50 = 34673685.05 nM T62449 C2Z6HW 49797814 IC50 = 39000 nM T62449 CM9BP3 49797815 IC50 > 100000 nM T62449 CNG4E3 49797838 IC50 = 30000 nM T62449 CX81ZB 49797839 IC50 = 13803842.65 nM T62449 CRQ74V 49797840 IC50 = 208000 nM T62449 CV7HS3 49797841 IC50 = 10000000 nM T62449 CWST49 49797842 IC50 = 10000000 nM T62449 CM2C5E 49797843 IC50 > 100000 nM T62449 C3GSC1 49797868 IC50 = 139000 nM T62449 C6X1YA 49797869 IC50 = 52000 nM T62449 CT4E9G 49797870 IC50 > 100000 nM T62449 CBHE98 49797871 IC50 = 5000 nM T62449 CO74EX 49797872 IC50 = 22000 nM T62449 CX5L4V 49797873 IC50 = 1500 nM T62449 C2I6WB 49797892 IC50 > 100000 nM T62449 C21OMN 49797893 IC50 = 46000 nM T62449 C7L9FX 49797894 IC50 = 23000 nM T62449 CNX17D 49797895 IC50 = 22000 nM T62449 C91CQL 49797896 IC50 > 100000 nM T62449 C2JN7M 49797915 IC50 = 10000000 nM T62449 C1S8UC 49797916 IC50 = 10000000 nM T62449 CJ92RE 49797917 IC50 = 38904514.5 nM T62449 C0AO7C 49797918 IC50 = 96000 nM T62449 C62UKI 49797936 IC50 = 25000 nM T62449 CYD82V 49797937 IC50 = 17000 nM T62449 C4EV8I 49797938 IC50 = 15000 nM T62449 CE6S0H 49797939 IC50 = 15000 nM T62449 CHSF07 49806372 IC50 > 1000 nM T62449 C75GBE 49837568 IC50 > 100000 nM T62449 CF91RS 49843531 IC50 > 10000 nM T62449 CX14RL 49864766 IC50 = 10 nM T62449 C41BRL 49864767 IC50 = 40 nM T62449 CDZ47Q 49864776 IC50 > 100 nM T62449 CFC5U2 49864777 IC50 > 100 nM T62449 CU90NP 49864778 IC50 > 100 nM T62449 CWA31I 49864779 IC50 > 100 nM T62449 CVM9L1 49864839 IC50 > 100 nM T62449 CXN87Z 49864840 IC50 > 100 nM T62449 CQU81Z 49865197 IC50 = 13.3 nM T62449 C6GZJ9 49865198 IC50 = 71.2 nM T62449 CKCE17 49865199 IC50 = 2.6 nM T62449 C7YN3R 49865256 IC50 = 10 nM T62449 CPT0G4 49865257 IC50 = 4.5 nM T62449 CZ5IR4 49865258 IC50 = 8.8 nM T62449 C8FPR3 49865259 IC50 = 3.7 nM T62449 C6XV8T 49865294 IC50 = 190 nM T62449 CI5ZS8 49865296 IC50 = 520 nM T62449 C5OVD3 49865297 IC50 = 10 nM T62449 C0G8TJ 49865298 IC50 = 30 nM T62449 C8TC4G 49865353 IC50 = 90 nM T62449 C3SH6Z 49865354 IC50 = 1590 nM T62449 CUKC68 49865355 IC50 = 60 nM T62449 CSC97L 49865357 IC50 = 210 nM T62449 C3NFM8 49865366 IC50 = 18.8 nM T62449 C8IU6J 49865367 IC50 > 100 nM T62449 C52MCY 49865402 IC50 = 20 nM T62449 CRL65C 49865403 IC50 = 100 nM T62449 CTR09U 49865404 IC50 = 24400 nM T62449 CV10JU 49865405 IC50 = 6 nM T62449 CA0V2L 49865416 IC50 = 7.6 nM T62449 CBV0N2 49865417 IC50 = 4.6 nM T62449 CL46XB 49865418 IC50 = 5.9 nM T62449 CF2E5Q 49865419 IC50 = 4.5 nM T62449 CW6ZC7 49865454 IC50 = 9 nM T62449 C64TKW 49865455 IC50 = 9 nM T62449 CA2G4J 49865456 IC50 = 40 nM T62449 CW4T0M 49865457 IC50 = 210 nM T62449 CA6G5B 49865458 IC50 = 3490 nM T62449 C5T6MK 49865464 IC50 = 8 nM T62449 CSDF82 49865493 IC50 = 40 nM T62449 C4SI8E 49865494 IC50 = 10 nM T62449 C58EUV 49865495 IC50 = 690 nM T62449 CO7UJ2 49865496 IC50 = 120 nM T62449 C91QJV 49865497 IC50 = 1590 nM T62449 C1DQ4B 49865508 IC50 = 0.8 nM T62449 C1GDV8 49865509 IC50 = 0.5 nM T62449 CU8VG1 49865510 IC50 > 100 nM T62449 CLM31B 49865511 IC50 = 33 nM T62449 CWH3V6 49865544 IC50 = 2960 nM T62449 C5PIT4 49865545 IC50 = 20 nM T62449 CKH58V 49865546 IC50 = 26 nM T62449 C2JO1C 49865547 IC50 = 160 nM T62449 C4ZP5F 49865561 IC50 = 78.9 nM T62449 CWV1N3 49865562 IC50 = 74.3 nM T62449 CMXR95 49865563 IC50 > 100 nM T62449 CQ79BT 49865564 IC50 = 64.9 nM T62449 C9WL0E 50925625 IC50 = 1 nM T62449 CO2EP4 50925626 IC50 = 1 nM T62449 C2Y6QS 50938552 IC50 > 10000 nM T62449 CAZQ43 51003133 IC50 = 7 nM T62449 C9NYP4 51036677 IC50 > 10000 nM T62449 C4WRY3 51037112 IC50 > 10000 nM T62449 CRI28Z 51037948 IC50 > 10000 nM T62449 CC40TE 52417176 IC50 = 684 nM T62449 CXA03W 52920796 IC50 = 200 nM T62449 CEQN27 52936621 Ki > 1000 nM T62449 CS0J7X 52941254 IC50 = 60 nM T62449 CI03NU 52941315 IC50 = 67 nM T62449 CS54GO 52941316 IC50 = 34 nM T62449 C0K9IP 52941333 IC50 = 5 nM T62449 C42TLG 52942464 IC50 = 5 nM T62449 C8FP9S 52942478 IC50 = 3 nM T62449 C16MLK 52942510 IC50 = 7 nM T62449 CJ0QF7 52943673 IC50 = 16 nM T62449 CF7YO4 52943706 IC50 = 292 nM T62449 CIX16P 52943707 IC50 = 60 nM T62449 CE1MH2 52943718 IC50 = 4 nM T62449 C74TGC 52944093 IC50 = 4 nM T62449 CBJ5W0 52944874 IC50 = 21 nM T62449 C2X3OF 52944876 IC50 = 19 nM T62449 CL92FD 52944910 IC50 = 14 nM T62449 CM0V8Y 52944911 IC50 = 5 nM T62449 CO46IN 52944963 IC50 = 8 nM T62449 CVS9T8 52944964 IC50 = 3 nM T62449 CUVC48 52945260 IC50 = 3 nM T62449 CN6X9R 52945980 IC50 = 9000 nM T62449 CC7H6J 52946058 IC50 = 2 nM T62449 C6QF3G 52946076 IC50 = 3 nM T62449 CFW69G 52946090 IC50 = 3 nM T62449 C9D1OF 52946123 IC50 = 9 nM T62449 CJ4N5R 52946126 IC50 = 2 nM T62449 C7LB8I 52946129 IC50 = 746 nM T62449 CZ4C3G 52946131 IC50 = 7 nM T62449 CAR06C 52946146 IC50 = 197 nM T62449 C71WEM 52946170 IC50 = 148 nM T62449 C7S9EC 52946171 IC50 = 211 nM T62449 CGEB92 52946191 IC50 = 27143 nM T62449 CFV2J5 52947335 IC50 = 4 nM T62449 C07ZAX 52947366 IC50 = 2 nM T62449 C8VO2S 52947369 IC50 = 707 nM T62449 CH2QO7 52947383 IC50 = 2 nM T62449 CG73LH 52948516 IC50 = 20 nM T62449 CDV43P 52948517 IC50 = 16 nM T62449 C18PAC 52948520 IC50 = 5 nM T62449 CXP7I1 52948521 IC50 = 4582 nM T62449 C2LY5H 52948522 IC50 = 9 nM T62449 CT41EG 52948563 IC50 = 4 nM T62449 C9ZD5X 52948594 IC50 = 3 nM T62449 C8QF7M 52948596 IC50 = 9 nM T62449 C4D3GF 52948601 IC50 = 937 nM T62449 CG23XB 52948639 IC50 = 24 nM T62449 CFZ9T4 52948643 IC50 = 56 nM T62449 CJ4C5A 52949738 IC50 = 2 nM T62449 COWY74 52949739 IC50 = 3 nM T62449 C0O9XA 52949803 IC50 = 9 nM T62449 CM9G3T 52949847 IC50 = 717 nM T62449 C6OTY5 53251320 IC50 > 18000 nM T62449 CCJ21O 53316780 IC50 = 45 nM T62449 CFR4O8 53317703 IC50 > 50000 nM T62449 CE8OY2 53317913 IC50 = 13 nM T62449 CY5QE4 53318087 IC50 = 2900 nM T62449 C9ML7Y 53318088 IC50 = 36000 nM T62449 C4UVQ1 53318089 IC50 > 50000 nM T62449 CE5A3Z 53318090 IC50 = 9400 nM T62449 C75YLI 53318091 IC50 = 5000 nM T62449 C3Q2EN 53319015 IC50 = 820 nM T62449 CQU59W 53319377 IC50 = 1000 nM T62449 CHY1P9 53319425 IC50 = 2100 nM T62449 CZO08F 53319426 IC50 = 280 nM T62449 CT18YA 53319427 IC50 = 1500 nM T62449 CJL16Z 53320317 IC50 = 5 nM T62449 CYC50X 53321363 IC50 = 480 nM T62449 CEA73G 53321632 IC50 = 60 nM T62449 CS80CN 53321968 IC50 = 28 nM T62449 C3RUA9 53322026 IC50 = 540 nM T62449 CT3E0R 53322964 IC50 = 26 nM T62449 CSF93R 53323279 IC50 = 104000 nM T62449 CU2DX3 53323332 IC50 = 6800 nM T62449 CTRG49 53323387 IC50 = 2000 nM T62449 CES3A7 53323388 IC50 = 140 nM T62449 CZ56QD 53324655 IC50 = 410 nM T62449 CJ5N7L 53324705 IC50 = 4000 nM T62449 C5A2QJ 53324706 IC50 = 87 nM T62449 CE4XD5 53324707 IC50 = 7 nM T62449 C9HO8U 53324708 IC50 = 70 nM T62449 C0SWQ7 53325960 IC50 = 860 nM T62449 CZ5A6E 53325961 IC50 = 51 nM T62449 C4BYP9 53325998 IC50 = 1080 nM T62449 C2VAO0 53326006 IC50 = 34 nM T62449 C9MC3A 53326007 IC50 = 7 nM T62449 COZ9M2 53326008 IC50 = 1700 nM T62449 CRMY65 53326009 IC50 = 290 nM T62449 CGE96S 53326873 IC50 = 35 nM T62449 COY19W 53326906 IC50 = 8 nM T62449 C0SWH5 53348216 IC50 > 40000 nM T62449 C8NA4L 53384644 IC50 > 30000 nM T62449 CVG90B 53389651 IC50 > 10000 nM T62449 CE1ZK6 54759168 IC50 > 10000 nM T62449 C8AB1J 54759606 Ki = 110 nM T62449 CXV2G6 54770686 IC50 > 100000 nM T62449 CES4B3 54770691 IC50 > 100000 nM T62449 C6Z2VS 54770693 IC50 > 100000 nM T62449 C3ZVT2 54770915 IC50 > 100000 nM T62449 CME94T 54771590 IC50 > 100000 nM T62449 C5GPT9 54771592 IC50 > 100000 nM T62449 C1TWQ3 54771822 IC50 > 100000 nM T62449 CBOD63 56835089 IC50 > 30000 nM T62449 C7DMC5 56926362 IC50 = 122000 nM T62449 C7VTR9 56926363 IC50 = 1200 nM T62449 C1DV2B 56932125 IC50 = 47 nM T62449 CAK91L 56955954 IC50 > 3600 nM T62449 CWX85I 57345537 IC50 = 10 nM T62449 CI70CT 57345538 IC50 = 20 nM T62449 CI82KP 57390271 IC50 > 100000 nM T62449 CHU67R 57390273 IC50 = 78500 nM T62449 C38TVB 57391918 IC50 = 3200 nM T62449 CT1ZU3 57391919 IC50 = 880 nM T62449 CE8T5V 57393795 IC50 = 13820 nM T62449 CM6F0O 57393798 IC50 > 100000 nM T62449 CGU57X 57394413 IC50 > 100000 nM T62449 CD6Y9Z 57395116 IC50 > 30000 nM T62449 C8W6IG 57395117 IC50 > 30000 nM T62449 CT9L8D 57395512 IC50 > 100000 nM T62449 CGU6C4 57395516 IC50 > 100000 nM T62449 CG7S0D 57396882 IC50 > 30000 nM T62449 CQ6Y4G 57397344 IC50 > 100000 nM T62449 CU1D3X 57400635 IC50 = 1500 nM T62449 C0UDY9 57401151 IC50 > 30000 nM T62449 CECL89 57402533 IC50 > 100000 nM T62449 C2VK6A 57404485 IC50 = 1.7 nM T62449 CK6T1C 57404486 IC50 = 0.07 nM T62449 CQ80BX 57404487 IC50 = 0.05 nM T62449 C48ATX 57752723 IC50 = 39 nM T62449 CR1B9I 57867443 IC50 = 19 nM T62449 C42IGJ 57867446 IC50 = 0.4 nM T62449 CO3L9P 57867459 IC50 = 350 nM T62449 CZ9CO1 57867473 IC50 = 6 nM T62449 C18QUW 57867482 IC50 = 27 nM T62449 CEXS06 57867488 IC50 = 113 nM T62449 CIZ91X 57867490 IC50 = 0.3 nM T62449 C1VFJ8 57867505 IC50 = 16 nM T62449 C3Z5KS 57867516 IC50 = 5 nM T62449 CFB7Q4 57867522 IC50 = 33 nM T62449 C31SCV 57867523 IC50 = 320 nM T62449 CDXQ72 58266334 EC50 = 95.8 nM T62449 CRZ21K 58266341 IC50 = 0.95 nM T62449 CV89NE 58266367 IC50 = 2.3 nM T62449 CL5H9F 58266371 EC50 = 540 nM T62449 C3BMF9 58266373 EC50 = 292 nM T62449 C54OAK 58266384 EC50 = 128 nM T62449 CGX93Z 58266397 IC50 = 4.2 nM T62449 CRP98K 58266398 EC50 = 339 nM T62449 CT9U4W 58266401 IC50 = 9.1 nM T62449 CKM8L7 58266405 IC50 = 18.6 nM T62449 C6RE1W 58266437 IC50 = 2.3 nM T62449 C8RVJ3 58266453 EC50 = 118 nM T62449 C85NFY 58266473 IC50 = 27.1 nM T62449 CMS4L5 58266501 IC50 = 38.1 nM T62449 CD0B2Y 58266522 IC50 = 127 nM T62449 CU2Q7N 58266536 EC50 = 2234 nM T62449 C0EZ8W 58266545 EC50 = 986 nM T62449 C3YB2K 58266559 IC50 = 4.1 nM T62449 CIY05G 58266579 EC50 = 23.9 nM T62449 CG5X8N 58266605 EC50 = 172 nM T62449 CO72RU 58266637 EC50 = 72.8 nM T62449 CAI4Q3 58266657 IC50 = 20.2 nM T62449 CA7Q9D 58266659 EC50 = 2495 nM T62449 CK6W9C 58266664 IC50 = 18.3 nM T62449 C6YJ2E 58266718 IC50 = 5.1 nM T62449 CKH57L 58266732 IC50 = 863 nM T62449 CL0F3T 58266741 IC50 = 1.8 nM T62449 C0MZH2 58266751 IC50 = 140 nM T62449 C89IKL 58266769 IC50 = 11.4 nM T62449 C8HT0J 58266791 IC50 = 0.31 nM T62449 CR3X6B 58266796 IC50 = 14.7 nM T62449 CT42VW 58266828 IC50 = 1.9 nM T62449 C6W7PQ 58266840 EC50 = 228 nM T62449 CW0Q6F 58902643 IC50 = 10 nM T62449 C0T7IJ 58902644 IC50 = 3 nM T62449 C6BPR2 58985201 IC50 > 30000 nM T62449 CT3EW2 59292007 IC50 = 950 nM T62449 CXO2D6 59331996 IC50 = 5200 nM T62449 CZ4R1I 59332136 IC50 = 281 nM T62449 C39FVZ 59332156 IC50 = 46 nM T62449 CNZG62 59332168 IC50 = 8 nM T62449 CGVA94 59332218 EC50 = 750 nM T62449 C4P6EW 59332249 EC50 = 75 nM T62449 C1I2ZJ 59332253 IC50 = 62 nM T62449 CA90ZE 59332270 IC50 = 10 nM T62449 C8QP2B 59332297 IC50 = 29 nM T62449 C12QIP 59332322 IC50 = 10000 nM T62449 COQ4G0 59332354 IC50 = 120 nM T62449 CT03UE 59332395 EC50 = 250 nM T62449 CP9A8T 59503659 IC50 = 300 nM T62449 C1MA6J 59503711 IC50 = 20 nM T62449 CX29EU 59503744 IC50 = 300 nM T62449 CXJ63M 59603829 IC50 = 190 nM T62449 CQEU96 59603842 IC50 = 2.2 nM T62449 C16YEO 59662448 IC50 > 50000 nM T62449 C1MR8Q 60097495 IC50 > 10000 nM T62449 C8MEP5 60155174 EC50 = 100 nM T62449 C6JG5S 60155175 IC50 = 13 nM T62449 C2FE5C 60155176 EC50 = 150 nM T62449 CZ2RH1 60155260 IC50 = 9 nM T62449 CR08WJ 60155261 EC50 = 20 nM T62449 C7ELC6 60155262 EC50 = 20 nM T62449 CE1LV8 60155263 IC50 = 40 nM T62449 C8VED4 60155264 EC50 = 40 nM T62449 CSZA16 60155724 IC50 > 3600 nM T62449 CK6WO0 66552478 IC50 < 10000 nM T62449 CBA0S2 66555775 IC50 = 232.5 nM T62449 CL1D5C 67076166 IC50 = 414 nM T62449 CZJG46 67203533 IC50 = 56.6 nM T62449 CV63UL 67240318 IC50 > 10000 nM T62449 C8CV4S 68346820 EC50 = 425 nM T62449 CXS64A 68502671 IC50 = 6800 nM T62449 CG6JX0 69010662 EC50 = 3300 nM T62449 CJ0QP9 69011075 IC50 = 140 nM T62449 C9SFL1 69011426 IC50 = 660 nM T62449 CDQ56Z 69011601 IC50 = 150 nM T62449 CYIB47 69012259 EC50 = 50 nM T62449 CF57OD 69012280 IC50 = 83 nM T62449 CG4L1J 69013144 EC50 = 390 nM T62449 CI8GH6 69013596 IC50 = 56 nM T62449 C5DGR9 69036886 IC50 = 10000 nM T62449 C3QMC9 69452020 IC50 = 20 nM T62449 CMPO35 69452226 IC50 = 10 nM T62449 C7FIO8 69452237 IC50 = 6 nM T62449 C8P1OC 69452405 IC50 = 40 nM T62449 CJ28CH 69453348 IC50 = 50 nM T62449 C53SLM 69453492 IC50 = 20 nM T62449 CB01WU 69453501 IC50 = 420 nM T62449 CH7D9T 69453726 IC50 = 30 nM T62449 CXR41C 69453775 IC50 = 9 nM T62449 CJG34E 69453791 IC50 = 10 nM T62449 CPS2I1 69453844 IC50 = 20 nM T62449 CF1JR8 69453892 IC50 = 600 nM T62449 CIO06M 69454063 IC50 = 30 nM T62449 C7V2BO 69454072 IC50 = 240 nM T62449 CT3FD4 69454764 IC50 = 4 nM T62449 C9N4WP 69454772 IC50 = 300 nM T62449 CD9HR5 69454819 IC50 = 20 nM T62449 C2YM6X 69454833 IC50 = 40 nM T62449 C9E8LF 69454898 IC50 = 400 nM T62449 C5H7SN 69455555 IC50 = 100 nM T62449 C7X3OP 69455815 IC50 = 20 nM T62449 C9J0NT 69455831 IC50 = 980 nM T62449 CU3YG5 69455856 IC50 = 5 nM T62449 CL4U5T 69455865 IC50 = 130 nM T62449 CMY31T 69455885 IC50 = 210 nM T62449 CK7OD5 69455944 IC50 = 300 nM T62449 C3F0ST 69456085 IC50 = 20 nM T62449 CA0Y7O 69456707 IC50 = 30 nM T62449 C0YG9L 69456717 IC50 = 160 nM T62449 C67POT 69456743 IC50 = 40 nM T62449 CS78TV 69457006 IC50 = 20 nM T62449 C4RH5P 69457015 IC50 = 30 nM T62449 CAC6Z2 69458213 IC50 = 850 nM T62449 C2C1TO 69458563 IC50 = 90 nM T62449 C65IOX 69458628 IC50 = 90 nM T62449 CPY64U 70680987 IC50 = 520 nM T62449 CM8LY4 70681104 IC50 = 12 nM T62449 CH46LV 70681807 IC50 = 4100 nM T62449 C16KCJ 70681808 IC50 > 50000 nM T62449 CA24BI 70681809 IC50 = 21000 nM T62449 CPG6A9 70681810 IC50 = 130 nM T62449 CY37AS 70681811 IC50 = 1400 nM T62449 C2H4GM 70682566 EC50 = 80 nM T62449 C8RI7V 70683114 IC50 = 0.27 nM T62449 C76BMR 70683916 IC50 > 50000 nM T62449 C7XUJ9 70683919 IC50 = 580 nM T62449 C9YTC5 70683920 IC50 = 520 nM T62449 CON6Q4 70683921 IC50 = 2000 nM T62449 C7ESU8 70684650 EC50 = 40 nM T62449 CSV7N6 70685303 IC50 = 110 nM T62449 CHC4P3 70685325 IC50 = 12 nM T62449 C7XGK0 70687350 IC50 = 440 nM T62449 CFJ6D0 70687445 IC50 = 440 nM T62449 CZIS95 70688169 IC50 = 4500 nM T62449 CCF0J9 70688170 IC50 = 760 nM T62449 CFA7X1 70688173 IC50 = 3400 nM T62449 C8UIF5 70688174 IC50 = 190 nM T62449 CR67KE 70688175 IC50 > 50000 nM T62449 CDZ45H 70690198 IC50 = 5200 nM T62449 C6QE8U 70690199 IC50 = 13000 nM T62449 CF0PE8 70691629 IC50 = 440 nM T62449 C49QWD 70691636 IC50 = 33 nM T62449 CB6Y5R 70692361 IC50 = 280 nM T62449 C1V8MZ 70692362 IC50 > 50000 nM T62449 CC7G4P 70692365 IC50 = 170 nM T62449 CR9E5Q 70692366 IC50 = 210 nM T62449 CQ3WS1 70692367 IC50 = 110 nM T62449 CZ60HX 70692368 IC50 = 190 nM T62449 CRE71P 70692369 IC50 = 1500 nM T62449 COE4K0 70693603 IC50 = 29 nM T62449 C9SK7N 70694424 IC50 > 50000 nM T62449 CD2HQ3 70694425 IC50 = 440 nM T62449 CJ95MK 70695151 IC50 = 6 nM T62449 CW2ME0 70695826 IC50 = 560 nM T62449 C0IA7J 70696492 IC50 = 3900 nM T62449 C5N2DQ 70697192 EC50 = 20 nM T62449 C4W9FY 70697193 EC50 = 30 nM T62449 C1IEJ2 70789254 IC50 = 18000 nM T62449 C8T7ZP 70789255 IC50 = 1800 nM T62449 CH0B8N 70789756 IC50 > 30000 nM T62449 C0NHM9 71098351 IC50 = 230 nM T62449 C6EKU0 71098352 IC50 = 870 nM T62449 C5LJ2R 71098462 IC50 = 4700 nM T62449 CQ41UR 71450379 IC50 = 135 nM T62449 C6DIL5 71450436 IC50 = 11 nM T62449 C5O6BN 71452202 IC50 < 1 nM T62449 C9AO0Q 71452203 IC50 = 6.3 nM T62449 C03DBO 71452204 IC50 = 7 nM T62449 CLE48V 71452268 IC50 = 36 nM T62449 CE0J5O 71454007 IC50 < 1 nM T62449 CB43OI 71454008 IC50 = 4.4 nM T62449 CG64AO 71454068 IC50 = 46.5 nM T62449 C8BRU5 71455750 IC50 = 110 nM T62449 CKT60L 71455860 Ki = 167 nM T62449 CMJ9N1 71457535 IC50 = 169 nM T62449 C6G3AS 71457582 IC50 = 18 nM T62449 C3IKX8 71457583 IC50 = 97 nM T62449 CFG21A 71459414 IC50 < 1 nM T62449 C1LIN4 71459486 IC50 = 21 nM T62449 CR2C6Z 71461172 IC50 = 5.4 nM T62449 CU9X6E 71461217 IC50 = 200 nM T62449 C5UB8I 71461218 IC50 = 10 nM T62449 CXE6H7 71461219 IC50 = 2.9 nM T62449 C6HN7D 71462955 IC50 = 20 nM T62449 CG2KF6 71462956 IC50 = 3.1 nM T62449 CCN01X 71547862 IC50 > 10000 nM T62449 CA3O6K 71552696 IC50 > 30000 nM T62449 C1NPL0 71552941 IC50 > 30000 nM T62449 CA4PS8 71552942 IC50 > 30000 nM T62449 C3UA9C 71553011 IC50 = 30000 nM T62449 CEZ15Y 71553012 IC50 = 30000 nM T62449 CVIA91 71553085 IC50 = 30000 nM T62449 C1TR3O 71553152 IC50 = 30000 nM T62449 CRX81Q 71575642 IC50 > 10000 nM T62449 CGE7S8 71602900 IC50 = 980 nM T62449 CY2M8J 71602948 EC50 = 1000 nM T62449 C08XIE 71614291 IC50 = 50000 nM T62449 CN1KE8 71614492 IC50 = 50000 nM T62449 CR4G1F 71614493 IC50 = 50000 nM T62449 CS57WM 72163974 IC50 = 12800 nM T62449 C06YGI 72165232 IC50 = 2 nM T62449 CB8ZU1 72188683 IC50 = 18 nM T62449 C9E4XZ 72546233 IC50 = 7100 nM T62449 C4B5RW 72725141 IC50 = 274 nM T62449 CY3U7T 73350434 IC50 = 42100 nM T62449 CSLQ67 76311610 IC50 = 45708818.96 nM T62449 CC82AE 76315190 IC50 = 10000000 nM T62449 CZ9NX5 76322493 IC50 = 10000000 nM T62449 C2Y4SD 76326091 IC50 = 45708818.96 nM T62449 C2H4LG 76326092 IC50 = 21877616.24 nM T62449 C6A9VB 76333357 IC50 = 43651583.22 nM T62449 CO0WJ9 86290236 IC50 = 1200 nM T62449 C0V8OG 86306050 IC50 = 123 nM T62449 C1HW4B 89735655 IC50 = 200 nM T62449 CFB75T 90479825 IC50 = 154 nM T62449 CY0UC4 90645194 IC50 > 10000 nM T62449 C0Y8ZK 91933875 IC50 > 1000 nM T62449 CAU45T 91971978 IC50 > 30000 nM T62449 CY7BI2 118706214 IC50 > 10000 nM T62449 CQX38N 118720611 IC50 = 44 nM T62449 CFP58Q 118720612 IC50 = 327 nM T62449 CF5HV8 118720613 IC50 = 80 nM T62449 C2UIB7 118720614 IC50 = 160 nM T62449 CSH50J 118720615 IC50 = 37 nM T62449 CYSD60 118720883 EC50 = 3300 nM T62449 C6E9UN 118720884 EC50 = 570 nM T62449 C4LW6I 118720885 IC50 = 80 nM T62449 C9Y4EH 118720886 IC50 = 84 nM T62449 C5Q2ZW 118720887 IC50 = 96 nM T62449 C3R9EN 118723883 IC50 = 1300 nM T62449 CQR9S1 118723884 IC50 = 4100 nM T62449 C9SH0Y 118723885 IC50 = 210 nM T62449 C5AP7D 118723886 IC50 = 60 nM T62449 CC50PY 118723887 IC50 = 390 nM T62449 CVPT50 118723888 IC50 = 1200 nM T62449 CQY17T 118723889 IC50 > 10000 nM T62449 C2X3OC 118723890 IC50 = 470 nM T62449 C86FOE 118723891 IC50 = 690 nM T62449 C62GMR 118723893 IC50 = 820 nM T62449 C1WFY9 118730799 IC50 = 26.57 nM T62449 CQC32W 118730800 IC50 = 9.9 nM T62449 CJ0IH1 118730801 IC50 = 21.55 nM T62449 CN6UX9 118730802 IC50 = 20.43 nM T62449 C05UZL 118730803 IC50 = 19.35 nM T62449 CTJG53 118730804 IC50 = 17.44 nM T62449 CQ48NV 118730805 IC50 = 15.54 nM T62449 C26OMX 118730806 IC50 = 13.63 nM T62449 CB47AL 118730807 IC50 = 12.78 nM T62449 CNTH27 118730808 IC50 = 11.89 nM T62449 CX50CM 118730809 IC50 = 22.64 nM T62449 CN26ZK 118730810 IC50 = 7.6 nM T62449 C2PT0H 118730811 IC50 = 1.65 nM T62449 CRUA27 118730812 IC50 = 4.59 nM T62449 CKJS86 118730813 IC50 = 3.48 nM T62449 CQYK51 118730814 IC50 = 2.57 nM T62449 CQCX41 118737057 IC50 > 10000 nM T62449 C9TSK8 122179405 IC50 = 16.6 nM T62449 C82GBW 122179406 IC50 = 76.5 nM T62449 C5JM8O 122179407 IC50 = 42.7 nM T62449 C4X7SD 122192466 IC50 > 10000 nM T62449 C93RQT 127038361 IC50 = 310 nM T62449 CHMT84 127038362 IC50 = 210 nM T62449 CVU8Z4 127038363 IC50 = 670 nM T62449 CB73NS 127038364 IC50 = 770 nM T62449 CJHQ62 127038729 IC50 = 530 nM T62449 CW4S0U 127039718 IC50 = 700 nM T62449 C8BSO6 127039719 IC50 = 990 nM T62449 CNH94T 127039720 IC50 = 540 nM T62449 C01LGZ 127039804 IC50 = 120 nM T62449 CYM0T6 127041396 IC50 = 800 nM T62449 CXM5Q6 127041397 IC50 = 800 nM T62449 CJI9D7 127041398 IC50 = 510 nM T62449 CGX1C5 127041399 IC50 = 910 nM T62449 C1G9QI 127042685 IC50 = 780 nM T62449 CZ3J4V 127042686 IC50 = 450 nM T62449 C27XTM 127042687 IC50 = 310 nM T62449 C0FM1R 130196825 IC50 = 9179 nM T62449 CJVT83 134507914 IC50 = 8.34 nM T62449 C08SZL 134507928 IC50 = 21.19 nM T62449 CY95HT 134507962 IC50 = 15.92 nM T62449 C21NSE 134507989 IC50 = 99.58 nM T62449 CRB72O 134507990 IC50 = 10.95 nM T62449 CKN6O8 134507992 IC50 = 12.71 nM T62449 CXT1A3 134508144 IC50 = 0.89 nM T62449 CK62QJ 134508152 IC50 = 1.96 nM T62449 CPD34I 134508190 IC50 = 4.72 nM T62449 CE9A3K 134508319 IC50 = 517.35 nM T62449 CC4LZ8 134508328 IC50 = 14.3 nM T62449 C6WS0K 135399706 IC50 = 1.4 nM T62449 CYO6W9 135399748 IC50 = 0.32 nM T62449 CS2LH3 135401179 IC50 = 0.35 nM T62449 CMVS34 135410282 IC50 = 731 nM T62449 C37ITY 135414445 IC50 = 62 nM T62449 C5AG7L 135414460 IC50 = 0.3 nM T62449 CK93CT 135418209 IC50 = 27 nM T62449 CQO3N9 135428146 IC50 > 30000 nM T62449 CU60YC 135431661 Ki = 0.36 nM T62449 CW0P1Q 135433657 IC50 = 237 nM T62449 C8X5SV 135433815 IC50 = 2950 nM T62449 CYN0G3 135435429 IC50 = 0.5 nM T62449 CLXB05 135438541 IC50 = 0.11 nM T62449 CD0IO6 135440394 Ki = 0.8 nM T62449 CT23XD 135444905 Ki = 50118.72 nM T62449 CV56JC 135451019 Ki = 0.38 nM T62449 CKJI53 135458230 IC50 = 6 nM T62449 CNWO10 135461992 Ki = 1.2 nM T62449 CDV6Z5 135464186 IC50 = 4.4 nM T62449 CR48OH 135468068 IC50 = 17 nM T62449 CJL78T 135469498 IC50 = 120 nM T62449 CF36ZX 135471783 IC50 = 100 nM T62449 CHE78N 135474408 IC50 = 7.7 nM T62449 CU5W1A 135487360 IC50 = 7.6 nM T62449 CPE67T 135487516 IC50 = 30 nM T62449 C9ABF8 135489323 IC50 = 3.3 nM T62449 C6K2VX 135489338 IC50 = 3.3 nM T62449 C52SOP 135499973 IC50 = 1373 nM T62449 CJ4V0A 135508121 IC50 = 0.25 nM T62449 CCKM76 135508625 IC50 = 66 nM T62449 C5L4HE 135511905 IC50 = 89 nM T62449 C4R5CG 135513005 IC50 = 1.04 nM T62449 CZE1Q5 135514607 Ki = 63.1 nM T62449 C2JA3F 135520167 IC50 = 0.3 nM T62449 CV5L0O 135525556 IC50 = 12 nM T62449 CF7DC6 135527483 IC50 = 24 nM T62449 C1F2TD 135559054 IC50 = 2.3 nM T62449 CMN71B 135559055 IC50 = 640 nM T62449 C25MKU 135559056 IC50 = 12 nM T62449 CHW54V 135559057 IC50 = 13 nM T62449 C4CJG9 135559058 IC50 = 80 nM T62449 CCQ4J8 135559059 IC50 = 10 nM T62449 CE6MF3 135559060 IC50 = 530 nM T62449 CDN21F 135559061 IC50 = 59 nM T62449 C8BJV6 135559062 IC50 = 12 nM T62449 CS4HA0 135559063 IC50 = 48 nM T62449 C2BHG0 135559064 IC50 = 2.6 nM T62449 CMF9Y8 135559065 IC50 = 30 nM T62449 C61XZP 135559066 IC50 = 110 nM T62449 CPC03V 135559067 IC50 = 34 nM T62449 C8G2TS 135559068 IC50 = 45 nM T62449 CTB7R2 135564980 IC50 = 85 nM T62449 C2LSE6 135566381 IC50 = 4500 nM T62449 CXW3V2 135566382 IC50 = 1070 nM T62449 CYN21W 135566732 IC50 = 25 nM T62449 C1FR5J 135566734 Ki = 3.981 nM T62449 C51DPR 135566735 Ki = 79.43 nM T62449 CW72QO 135580408 IC50 > 100000 nM T62449 CK3H9X 135582730 Ki = 79.43 nM T62449 CRJ45X 135589980 IC50 = 6.2 nM T62449 C2NMK7 135616966 IC50 = 0.1 nM T62449 C0J3BN 135678111 IC50 = 18 nM T62449 C70XQR 135742188 IC50 = 40 nM T62449 CX6D7L 135779185 Ki = 79.43 nM T62449 C3QF1W 135796851 IC50 = 0.24 nM T62449 C97MNL 135796852 IC50 = 9.3 nM T62449 C0HRJ6 135839313 Ki = 301 nM T62449 C9PM0V 135908179 IC50 = 0.74 nM T62449 CQ60FT 135908180 EC50 = 880 nM T62449 C83ATO 135908184 EC50 = 1300 nM T62449 CZV1F2 135921336 IC50 = 990 nM T62449 C8GU3S 135921380 IC50 = 20500 nM T62449 CN8PE1 135921414 IC50 = 1320 nM T62449 CO4HB9 135921450 IC50 = 26000 nM T62449 C35LMX 135921456 IC50 = 1100 nM T62449 C1JPV8 135921468 IC50 = 850 nM T62449 C6NPJ1 135921474 IC50 = 870 nM T62449 C5ID4X 135921475 IC50 = 200 nM T62449 CF96QY 135921485 IC50 = 870 nM T62449 C84AKH 135921502 IC50 = 1750 nM T62449 C0V8ZL 135921504 IC50 = 56000 nM T62449 C6GZC8 135921505 IC50 = 28000 nM T62449 C8SD7O 135921523 IC50 = 27500 nM T62449 CL67HX 135921546 IC50 = 140 nM T62449 CHI61Y 135926123 IC50 = 29 nM T62449 C3IS7L 135926124 IC50 = 14 nM T62449 CEQ5A7 135950133 IC50 = 3600 nM T62449 CH32XK 135955268 IC50 = 640 nM T62449 CA3YO7 135955269 IC50 = 16 nM T62449 C7F4LO 135965980 Ki = 3.981 nM T62449 CT54OI 135966023 Ki = 251.19 nM T62449 CS28HU 135966024 Ki = 7943.28 nM T62449 C43NXR 135966026 Ki = 398.11 nM T62449 CWX7G3 135966065 IC50 = 124 nM T62449 CHTU98 135966067 Ki = 0.5012 nM T62449 C1SI4P 135966068 Ki = 1995.26 nM T62449 C4GVZ2 135988232 IC50 = 29 nM T62449 C4L2ZH 135999903 IC50 = 130 nM T62449 CHA4N2 136013680 IC50 > 10 nM T62449 C6BLT4 136016455 IC50 = 43000 nM T62449 C8T5ZB 136016456 IC50 = 6500 nM T62449 CA5IK3 136020049 IC50 = 1554 nM T62449 C5XIE8 136026041 IC50 = 24000 nM T62449 CD56MA 136030632 IC50 = 260 nM T62449 C9IYG7 136030656 IC50 = 2600 nM T62449 CD5N4W 136030657 IC50 = 5050 nM T62449 CSJM98 136030658 IC50 = 230 nM T62449 CBT1R7 136034784 Ki = 0.18 nM T62449 C6SZH8 136034785 Ki = 0.2 nM T62449 CXGZ47 136034786 Ki = 0.3 nM T62449 COC4T2 136042307 IC50 = 1310 nM T62449 C0F7XG 136042308 IC50 = 867 nM T62449 CG4S3N 136042309 IC50 = 905 nM T62449 CSV49P 136042310 IC50 > 10000 nM T62449 CU4FI9 136042311 IC50 > 10000 nM T62449 CF5S9E 136042312 IC50 > 10000 nM T62449 CT4VZ5 136042313 IC50 > 10000 nM T62449 CQ69XH 136042314 IC50 = 6558 nM T62449 CV71CS 136044168 IC50 < 100 nM T62449 C13VUJ 136048734 Ki = 316.23 nM T62449 C62FHT 136059697 IC50 = 140 nM T62449 CZA3S5 136059698 IC50 = 890 nM T62449 CXP7U8 136059699 IC50 = 460 nM T62449 CF0T6L 136059700 IC50 > 10000 nM T62449 CD8S7G 136059701 IC50 > 10000 nM T62449 CVP95B 136059702 IC50 = 260 nM T62449 CJF74C 136059703 IC50 = 1700 nM T62449 C9I3AT 136059704 IC50 = 150 nM T62449 C2WQ1E 136059705 IC50 = 1300 nM T62449 C8LWQ3 136059706 IC50 = 230 nM T62449 C42QMW 136059707 IC50 = 180 nM T62449 C5B0YX 136059708 IC50 = 190 nM T62449 C6NGR5 136059709 IC50 = 280 nM T62449 CQKX19 136059710 IC50 > 10000 nM T62449 CWSJ54 136059711 IC50 > 10000 nM T62449 CIA81M 136059712 IC50 = 150 nM T62449 CVPZ19 136059713 IC50 = 300 nM T62449 CXGE05 136060550 EC50 = 4700 nM T62449 C5KF8E 136060551 IC50 = 6.6 nM T62449 C45SFB 136060552 IC50 = 3.9 nM T62449 C0WOE5 136060553 EC50 = 4000 nM T62449 C9E5RJ 136060554 IC50 = 4 nM T62449 C26ESH 136060555 IC50 = 13 nM T62449 C3L9MY 136060556 IC50 = 3.6 nM T62449 CMQV16 136060596 IC50 = 24 nM T62449 CC1AL2 136060597 IC50 = 6.4 nM T62449 C0JZ7V 136060598 IC50 = 1.2 nM T62449 CO40QX 136060599 IC50 = 2.1 nM T62449 C80NBR 136060600 IC50 = 0.74 nM T62449 C4SBU2 136060601 IC50 = 5.5 nM T62449 C29OYL 136060602 IC50 = 7.8 nM T62449 CUED80 136060603 IC50 = 209 nM T62449 CW69XL 136060604 IC50 > 10000 nM T62449 C3EA8H 136060605 IC50 > 10000 nM T62449 C1AFT3 136060606 IC50 = 34 nM T62449 C0F7MC 136060607 IC50 = 12 nM T62449 CN05HT 136060608 IC50 = 5.2 nM T62449 CBL4X6 136060609 IC50 = 7.1 nM T62449 CUMF79 136060610 IC50 = 5 nM T62449 C0NIC4 136060611 IC50 = 2.3 nM T62449 C8Z4ED 136060612 IC50 = 91 nM T62449 CU6B4P 136060613 IC50 = 671 nM T62449 CI43CY 136060614 IC50 = 0.24 nM T62449 C4W8FM 136060615 IC50 = 2.3 nM T62449 C9K3MC 136060616 IC50 = 0.83 nM T62449 C3XK6H 136060617 IC50 = 0.55 nM T62449 C8MYK4 136060618 IC50 = 0.43 nM T62449 CMD4J8 136060619 IC50 = 0.51 nM T62449 CK9TP4 136060620 IC50 = 0.21 nM T62449 CT32JA 136060621 IC50 = 0.56 nM T62449 CK48AB 136060622 IC50 = 1.1 nM T62449 C3KND8 136060623 IC50 = 18 nM T62449 C3EVB5 136060624 IC50 = 27 nM T62449 CDTB41 136060625 IC50 = 9091 nM T62449 C0VY4I 136060626 IC50 = 28 nM T62449 C15EDV 136060627 IC50 > 10000 nM T62449 C7ZIF0 136068426 IC50 = 330 nM T62449 C9S4LY 136068463 IC50 = 1700 nM T62449 C8DG4N 136068480 IC50 = 105 nM T62449 CC9U6S 136068516 IC50 = 4650 nM T62449 C1M6BD 136068537 IC50 = 1910 nM T62449 CWZX19 136087129 IC50 = 24.73 nM T62449 CD3U6W 136087130 IC50 = 7.54 nM T62449 CR1S9M 136087131 IC50 = 23.2 nM T62449 C7AQ9X 136087132 IC50 = 9.84 nM T62449 C9GMP3 136087133 IC50 = 5.36 nM T62449 CD1HY8 136087134 IC50 = 2.33 nM T62449 C49VON 136087135 IC50 = 15.34 nM T62449 C3UOC4 136087136 IC50 = 4.83 nM T62449 CG2VJ6 136087137 IC50 = 6.23 nM T62449 C26IDC 136087138 IC50 = 40.98 nM T62449 CL6J4F 136087139 IC50 = 3.53 nM T62449 C7A5SC 136087140 IC50 = 4.05 nM T62449 CG6YZ7 136087141 IC50 > 10000 nM T62449 C3MS1T 136087142 IC50 > 10000 nM T62449 CB36QU 136087143 IC50 > 10000 nM T62449 CW4VC1 136087144 IC50 > 10000 nM T62449 C2B4YQ 136087145 IC50 > 10000 nM T62449 C54DIE 136087146 IC50 > 10000 nM T62449 C4SDZ1 136087147 IC50 = 177.8 nM T62449 CA3D4R 136087148 IC50 > 10000 nM T62449 CA4J9I 136087149 IC50 > 10000 nM T62449 CL8B9K 136087150 IC50 = 116.1 nM T62449 CF0ME5 136087151 IC50 > 10000 nM T62449 C2MDW3 136087152 IC50 = 14.02 nM T62449 CE6OC8 136087153 IC50 = 9.94 nM T62449 C2EN1V 136087154 IC50 = 47.5 nM T62449 CI97YR 136087155 IC50 = 5.22 nM T62449 CG05JU 136087156 IC50 = 15.6 nM T62449 C4H8RT 136094854 IC50 = 138 nM T62449 C26WVM 136094855 IC50 = 482 nM T62449 CGF6L0 136094856 IC50 = 21.7 nM T62449 CL4F2M 136094857 IC50 = 7.2 nM T62449 C36YIP 136104482 IC50 = 1980 nM T62449 CYK85S 136104483 IC50 = 1370 nM T62449 CJAR29 136104484 IC50 = 7080 nM T62449 CK3J6B 136104485 IC50 = 230 nM T62449 C5AUZ1 136104486 IC50 = 1490 nM T62449 CNHJ52 136104487 IC50 = 58 nM T62449 CYZ08M 136104488 IC50 = 28860 nM T62449 CZ1WP6 136104489 IC50 = 290 nM T62449 C0BVF7 136104490 IC50 > 100000 nM T62449 C67WYQ 136104496 Ki = 0.2512 nM T62449 CBK18Q 136104497 IC50 = 2 nM T62449 C9UD4O 136104498 Ki = 0.19 nM T62449 CRU4W5 136104499 Ki = 0.5 nM T62449 C4GVM2 136104500 IC50 = 0.3 nM T62449 C5D6QJ 136104501 IC50 = 0.3 nM T62449 CG3K7Y 136118036 IC50 = 2 nM T62449 CF6M8A 136118037 IC50 = 74 nM T62449 CDZC97 136118038 IC50 = 5 nM T62449 CHN93K 136118039 IC50 = 0.8 nM T62449 CM25BJ 136118040 Ki = 0.1 nM T62449 C2KMO0 136118041 IC50 = 5 nM T62449 CT30HK 136118042 IC50 = 30 nM T62449 CDE5U4 136118043 IC50 = 0.8 nM T62449 C4L7HR 136118044 IC50 = 4 nM T62449 CDK61I 136118045 IC50 = 23 nM T62449 CGZ4K7 136118046 IC50 = 3 nM T62449 CP3E9H 136118047 IC50 = 5 nM T62449 C0IRU1 136118048 IC50 = 2 nM T62449 C9A7MH 136118049 IC50 = 290 nM T62449 C3W2HJ 136118050 IC50 = 62 nM T62449 CYV6H0 136118051 IC50 = 21 nM T62449 C4WY5K 136118052 IC50 = 0.1 nM T62449 CBR7H1 136118053 IC50 = 2 nM T62449 CT3VQ6 136118054 IC50 = 0.7 nM T62449 CI4E9L 136118055 Ki = 1.585 nM T62449 CN9TZ1 136118056 IC50 = 5 nM T62449 CQ5B6D 136118057 IC50 = 18 nM T62449 CUAV21 136118058 IC50 = 0.4 nM T62449 C4LTW8 136118059 IC50 = 23 nM T62449 CD8QK7 136118060 IC50 = 1 nM T62449 CK28XC 136118061 IC50 = 36 nM T62449 CQ91LF 136118062 IC50 = 24 nM T62449 CN4VG5 136118063 IC50 = 0.6 nM T62449 CFB7N4 136118064 IC50 = 0.6 nM T62449 CSTQ81 136118065 IC50 = 20 nM T62449 CAC8I4 136118066 IC50 = 8 nM T62449 C0OU2L 136118067 IC50 = 2 nM T62449 CA1KS3 136118068 IC50 = 0.8 nM T62449 CF2N3L 136118069 IC50 = 10 nM T62449 CTV6L5 136118070 IC50 = 8 nM T62449 CEGI81 136118071 IC50 = 40 nM T62449 CY9Q5S 136118072 IC50 = 0.2 nM T62449 C8GPW6 136118073 IC50 = 0.7 nM T62449 C45GKH 136118074 IC50 = 25 nM T62449 CP0NI8 136118075 IC50 = 6 nM T62449 C6AGD3 136118076 IC50 = 2 nM T62449 C4VI8W 136118077 IC50 = 1 nM T62449 CPYS69 136118078 IC50 = 2 nM T62449 C0O3WY 136118079 IC50 = 13 nM T62449 CHF4X3 136118080 IC50 = 0.2 nM T62449 C96NJX 136118081 IC50 = 0.8 nM T62449 C1CJ7W 136118082 IC50 = 48 nM T62449 CN36GJ 136118083 IC50 = 2 nM T62449 C4GRS6 136123435 Ki = 39.81 nM T62449 CKA48P 136123465 Ki = 501.19 nM T62449 C25ADI 136127009 IC50 = 50 nM T62449 CZ7EX0 136183413 IC50 = 5940 nM T62449 C1YUD0 136219394 IC50 > 10 nM T62449 COG2M5 136242661 Ki = 10 nM T62449 C9S7HU 136254220 IC50 = 100 nM T62449 C5ACT7 136254221 IC50 = 1200 nM T62449 CIU8W3 136254389 IC50 > 10 nM T62449 C83WAK 137189946 IC50 = 690 nM T62449 C8KW0I 137189951 IC50 = 750 nM T62449 COX23B 137189952 IC50 = 560 nM T62449 C04YDK 137248544 Ki = 7 nM T62449 CMB78I 137301774 Ki = 81 nM T62449 C0H5DU 137634144 IC50 = 6 nM T62449 C8GQD5 137636872 IC50 = 57 nM T62449 CC1Y6W 137645554 EC50 = 410 nM T62449 C1PSL6 137647194 IC50 = 2600 nM T62449 CZ89GD 137651664 IC50 = 79 nM T62449 C9Z1HL 137653065 EC50 = 2300 nM T62449 CO9SD0 137654952 EC50 = 10 nM T62449 CW24JK 137656651 EC50 = 10000 nM T62449 C8YB3D 137657887 EC50 = 30 nM T62449 CHQA31 138454800 IC50 = 0.4 nM T62449 C6VB3O 145925651 IC50 >= 5000 nM T62449 CGJ51K 145951051 IC50 = 8060 nM T62449 CYE53Z 145954734 IC50 = 9870 nM T62449 CT3GD2 145956060 IC50 = 2570 nM T62449 CO4JX8 145957090 IC50 = 1270 nM T62449 CDNC31 145967951 IC50 = 13 nM T62449 CHLZ93 145971754 IC50 = 3630 nM T62449 C3DJ7Z 145973152 IC50 = 3600 nM T62449 C3C9MT 145974327 IC50 = 2830 nM T62449 C8G5IE 145986785 IC50 = 1300 nM T62449 C2MD1Q 155513187 IC50 > 10000 nM T62449 CV4RX3 155514202 IC50 = 26.3 nM T62449 C3EW5X 155515884 IC50 = 6053.5 nM T62449 CKIB47 155516367 IC50 = 2.58 nM T62449 CG6PI4 155517225 IC50 = 0.5 nM T62449 CVA09Y 155517475 IC50 = 26.33 nM T62449 CSUR84 155518803 IC50 = 19.43 nM T62449 CUC01N 155522751 IC50 = 58.94 nM T62449 C1AJ7D 155524995 IC50 = 1.8 nM T62449 C9T1YO 155531676 IC50 = 4.49 nM T62449 CCDX27 155532778 IC50 = 1406 nM T62449 C6KTQ5 155534319 IC50 = 1.3 nM T62449 CZ8LG6 155536329 IC50 = 29.02 nM T62449 CV38WN 155536800 IC50 = 1.43 nM T62449 C3LC9I 155536820 IC50 = 1584.89 nM T62449 CFO2D3 155539849 IC50 = 4.72 nM T62449 CIKQ62 155541387 IC50 = 8.88 nM T62449 C57DTS 155549167 IC50 = 1610 nM T62449 CO0Q7V 155551803 IC50 = 8.76 nM T62449 CZQM57 155554194 IC50 = 0.4 nM T62449 C0H4KR 155555210 IC50 = 15.14 nM T62449 CC47VI 155556409 IC50 = 6.44 nM T62449 CLT5A0 155556574 IC50 = 365.25 nM T62449 CBA48E 155558852 IC50 = 3.75 nM T62449 C6IO8W 155559462 IC50 = 2.43 nM T62449 CTSK16 155562596 IC50 = 3.62 nM T62449 CIE3G4 155566394 IC50 = 59.49 nM T62449 CYZ63I 155566717 IC50 = 2.56 nM T62449 CG90RD 45267008 Ki = 501.19 nM T62449 CEZ6R1 45271206 Ki = 1.995 nM T62449 CR7LH1 9881974 Ki = 15848.93 nM T62449 D00ERW 44444843 Ki = 4 nM T62449 D00HVA 11624601 Ki > 8800 nM T62449 D00KDF 3387354 IC50 = 15 nM T62449 D01HUO 10086414 IC50 = 20 nM T62449 D01WAI 135451156 IC50 = 330 nM T62449 D03DZO 11715767 IC50 > 10000 nM T62449 D04ZWF 53396311 IC50 > 10000 nM T62449 D06EZQ 5324595 IC50 = 81 nM T62449 D08HFG 24809764 IC50 > 10000 nM T62449 D09HVH 135566652 IC50 > 10 nM T62449 D09YHQ 11993732 IC50 = 580 nM T62449 D09YVU 44443516 IC50 = 98 nM T62449 D0CM6T 11314340 Ki = 2600 nM T62449 D0D6DH 10125830 IC50 = 7 nM T62449 D0DH1H 135564841 IC50 = 190 nM T62449 D0F0AX 135413546 IC50 = 1950 nM T62449 D0FO2K 848641 IC50 = 22900 nM T62449 D0K0UJ 49837564 IC50 > 100000 nM T62449 D0M9OF 5329371 IC50 = 1000 nM T62449 D0ME9B 46868971 IC50 = 140 nM T62449 D0O6OH 71553154 IC50 = 1370 nM T62449 D0Q3KS 9957049 IC50 > 10000 nM T62449 D0Q3NG 11715520 Ki > 8800 nM T62449 D0S3TJ 76098 IC50 = 42000 nM T62449 D0S7IE 11658882 Ki > 8800 nM T62449 D0T8NU 16757525 IC50 > 4000 nM T62449 D0W7TU 947057 IC50 > 50000 nM T62449 D0Y3PH 11844342 IC50 = 470 nM T62449 D0Y5RO 4566 IC50 < 500 nM T62449 D0Z2CN 135418335 IC50 = 100 nM T62449 D0Z8PT 54758482 IC50 = 7.7 nM T97136 D03LWG 53235510 IC50 > 10000 nM T97136 D06EGV 44603533 IC50 = 130 nM T97136 D07EHV 44814409 IC50 > 10000 nM T97136 D07XOV 118598754 IC50 = 2.4 nM T97136 D0E3TC 44259 IC50 = 52.7 nM T97136 D0ZH4I 76071870 IC50 = 570 nM T97136 D0Q7HO 4705 IC50 = 630 nM T97136 CH21PG 2428 IC50 = 2800 nM T97136 CMB1E7 3796 IC50 = 120 nM T97136 C1ACH4 255690 IC50 = 580 nM T97136 CVQ15R 459521 IC50 = 14000 nM T97136 C6QKU7 711496 IC50 = 1350 nM T97136 C1DJU8 713705 IC50 = 2180 nM T97136 C6OI7A 713708 IC50 = 1620 nM T97136 C19AIM 713716 IC50 = 1790 nM T97136 C63CDO 756646 IC50 = 850 nM T97136 CRP8Y4 831273 IC50 = 2430 nM T97136 C7B9CV 932209 IC50 = 1560 nM T97136 CAX35I 1103000 IC50 = 1510 nM T97136 CN1AT4 1400686 IC50 = 1700 nM T97136 C2Y9UB 1515243 IC50 = 35000 nM T97136 CK5WN4 1515244 IC50 = 31000 nM T97136 C15MJS 2239542 Ki > 10000 nM T97136 C6JES2 2421499 IC50 = 1090 nM T97136 C8SYF6 2725997 IC50 = 27000 nM T97136 CI9N4S 2735305 IC50 = 62000 nM T97136 CJGT05 2735393 IC50 = 103000 nM T97136 C6R5VD 2735821 IC50 = 76000 nM T97136 CPI2C5 2775690 IC50 = 180000 nM T97136 CE16XS 2780715 IC50 = 50000 nM T97136 CU0V1A 4739100 IC50 = 10000 nM T97136 CS52EI 5047828 IC50 = 160 nM T97136 C4RUV5 5329453 IC50 = 130 nM T97136 CD06PU 9878588 IC50 = 3800 nM T97136 CVN8T9 10379252 IC50 = 120 nM T97136 C8E4TS 11992146 IC50 > 10000 nM T97136 CJR7W4 13521419 IC50 = 700 nM T97136 CD1I7O 14623308 Ki = 507 nM T97136 CUR7H3 16719862 IC50 = 16000 nM T97136 C38FDZ 16760660 IC50 = 120 nM T97136 CDMI50 23661564 IC50 > 200000 nM T97136 CZ25YH 24821077 IC50 = 5150 nM T97136 CR2W7S 28855509 Ki = 1900 nM T97136 CZ63DC 39817743 IC50 = 3000 nM T97136 CLI16E 44465026 IC50 = 20000 nM T97136 CQ7W3Y 46182043 Ki > 10000 nM T97136 CQJ1W7 46182661 Ki = 186 nM T97136 C08EBI 46937430 IC50 = 646 nM T97136 CQ3KU9 50899556 IC50 = 45 nM T97136 C3LB5V 52941849 IC50 = 2200 nM T97136 CTFK37 52941940 IC50 = 4050 nM T97136 C1HZ0B 52941952 IC50 = 1710 nM T97136 CD1G9Y 52942025 IC50 = 3240 nM T97136 CY70KP 52943231 IC50 = 4280 nM T97136 CW2X5E 52944268 IC50 = 950 nM T97136 CGZA67 52944340 IC50 = 1530 nM T97136 C0IAJ5 52945438 IC50 = 2930 nM T97136 CY6FK5 52945599 IC50 = 6180 nM T97136 CPI7U4 52945661 IC50 = 1620 nM T97136 CEW9P3 52945662 IC50 = 2410 nM T97136 C9PX2J 52945752 IC50 = 27 nM T97136 CL4ED3 52945753 IC50 = 164 nM T97136 CD2S4X 52946794 IC50 = 1800 nM T97136 CIR3Q0 52947964 IC50 = 1100 nM T97136 CPA63Q 52949333 IC50 = 4090 nM T97136 C1XS2J 54760383 IC50 = 6700 nM T97136 CV56NF 57428036 IC50 = 8800 nM T97136 CI10DA 58452049 IC50 = 292000 nM T97136 CIYE78 59225955 IC50 = 690 nM T97136 CV63UL 67240318 IC50 > 10000 nM T97136 CRF2P7 68233509 Ki > 10000 nM T97136 CH45ZR 71744719 IC50 = 23 nM T97136 C8YA3T 71766208 IC50 = 9 nM T97136 C5CDM4 71766212 IC50 = 570 nM T97136 C6P9HZ 71766360 IC50 = 64 nM T97136 C24OTM 72191544 IC50 = 1 nM T97136 C46WQC 72548802 IC50 = 5 nM T97136 C2PAK9 73438493 IC50 = 200 nM T97136 CHI51J 76070594 IC50 = 5680 nM T97136 C8VAD5 76070929 IC50 = 350 nM T97136 CB4V1R 76071142 IC50 = 5980 nM T97136 CBAT06 76071144 IC50 = 2520 nM T97136 C7SH1T 76071506 IC50 = 510 nM T97136 CS87EI 76071624 IC50 = 3920 nM T97136 CGC0K4 76071869 IC50 = 350 nM T97136 CGD0S5 89825760 IC50 = 84 nM T97136 CR5H9I 89826764 IC50 = 369 nM T97136 C7GC8K 89826796 IC50 = 238 nM T97136 C1IA0Q 89826982 IC50 = 20 nM T97136 CMJY71 89827041 IC50 = 499 nM T97136 CT6W0Y 89835558 IC50 = 16 nM T97136 C5VAT0 90024584 IC50 = 6 nM T97136 CG7YI5 90167717 IC50 = 170000 nM T97136 CBP5K7 91183030 IC50 = 3690 nM T97136 CDM21G 117737362 IC50 = 574 nM T97136 CWL6D7 117737365 IC50 = 331 nM T97136 CZK36G 118062095 IC50 = 3540 nM T97136 C07FTJ 118062454 IC50 = 6 nM T97136 CR6G8P 118242667 Ki > 10000 nM T97136 C01HYG 118598634 IC50 = 3.3 nM T97136 CL5W7Y 118598693 IC50 = 0.51 nM T97136 C9F0JN 118598698 IC50 = 2.7 nM T97136 C2KW9T 118598721 IC50 = 60 nM T97136 CDSW54 118598782 Ki = 2 nM T97136 C2MI8L 118598816 IC50 = 0.65 nM T97136 CL0Q6D 118598855 IC50 = 2 nM T97136 C1X9MR 118598890 IC50 = 1.4 nM T97136 C71FQV 118598955 IC50 = 10 nM T97136 C48RSO 118598997 IC50 = 2.2 nM T97136 CCB0Q3 118599016 IC50 = 0.88 nM T97136 C4OZ3A 118599023 IC50 = 1.6 nM T97136 C6BEH9 118599128 IC50 = 6.5 nM T97136 CN0BQ3 118734651 Ki > 10000 nM T97136 C1U0RH 118734652 Ki > 10000 nM T97136 C1UTE7 118734653 Ki = 4820 nM T97136 COK64U 118734654 Ki = 2060 nM T97136 C6WQT5 118734655 Ki > 10000 nM T97136 C5ZD2P 118734656 Ki > 10000 nM T97136 C2LBN0 118734657 Ki > 10000 nM T97136 CIR0W7 118734658 Ki = 5400 nM T97136 CS6GO0 118734659 Ki = 5000 nM T97136 CJ5KP0 118734660 Ki = 2330 nM T97136 C3CFZ7 118734661 Ki > 10000 nM T97136 CN0Z5J 118734662 Ki = 2150 nM T97136 C7ZN0X 118734663 Ki = 4510 nM T97136 CC2T5L 121007996 IC50 = 42000 nM T97136 CC4P7E 122194697 Ki = 1020 nM T97136 CH3BN2 122194698 Ki = 106 nM T97136 CGD5E3 122194699 Ki = 933 nM T97136 CYR1F2 122194700 Ki > 10000 nM T97136 C7YMU6 122194701 Ki = 320 nM T97136 C8DW9G 122485490 IC50 = 2680 nM T97136 C4PFZ0 127046319 IC50 = 36 nM T97136 C0CX4P 127046320 IC50 = 4 nM T97136 CUD8G5 127046367 IC50 = 80 nM T97136 CA83YU 127047442 IC50 = 2 nM T97136 CNJQ71 127047443 IC50 = 1.5 nM T97136 CC1VO7 127047444 IC50 = 3 nM T97136 C3IRJ0 127048197 IC50 > 10000 nM T97136 CZ07TW 127048198 IC50 > 10000 nM T97136 CS0H2C 127048199 IC50 > 10000 nM T97136 C1OE2F 127049532 IC50 = 370 nM T97136 C5P8TC 127049857 IC50 > 10000 nM T97136 CPQ35R 127049870 IC50 = 540 nM T97136 CQO3X7 127049871 IC50 > 10000 nM T97136 C5H8LK 127051998 IC50 > 10000 nM T97136 CGT0B1 127052321 IC50 = 7700 nM T97136 C7NH6A 127052914 IC50 > 10000 nM T97136 CKB1Y6 127052915 IC50 = 4510 nM T97136 C3B8RF 129071308 IC50 = 28 nM T97136 CN3K0W 129071500 IC50 = 23 nM T97136 CJ71ME 129071521 IC50 = 100 nM T97136 CZ5TU6 129071545 IC50 = 1.9 nM T97136 C1UWQ9 129956867 IC50 = 34000 nM T97136 CH8DP7 132220479 IC50 = 66 nM T97136 C8MQ2S 135471989 IC50 = 8170 nM T97136 CJF28E 136273088 IC50 = 125 nM T97136 CXY09A 136621908 IC50 = 60 nM T97136 C4L5AY 136623815 IC50 = 284 nM T97136 C6YQ4P 137349311 IC50 = 6400 nM T97136 CLV25F 137631507 IC50 = 3000 nM T97136 CQR0I4 137637598 IC50 = 4700 nM T97136 C9ZO5R 137652825 IC50 = 1.5 nM T97136 C5G7EA 139307786 IC50 = 600 nM T97136 CXHK68 140999007 IC50 = 61000 nM T97136 CSG67A 141009064 IC50 = 236000 nM T97136 CL5F4T 141381328 IC50 = 528 nM T97136 CU65MQ 145915878 IC50 = 800 nM T97136 CNK29G 145949498 Ki = 4770 nM T97136 CFV8U4 145952625 Ki = 890 nM T97136 CV8DJ4 145952962 Ki = 5920 nM T97136 CM1XY4 145954013 Ki = 1770 nM T97136 CMY39G 145956109 Ki = 940 nM T97136 CR8O6B 145956516 Ki = 860 nM T97136 C6D0NW 145956852 Ki = 710 nM T97136 CEK3W0 145958852 Ki = 1310 nM T97136 C3N1XY 145959793 Ki = 1470 nM T97136 CM8ZA1 145960224 Ki = 1230 nM T97136 CXU0Z9 145964697 IC50 = 224 nM T97136 CR7HU3 145964902 IC50 = 789 nM T97136 C42FZC 145966011 IC50 = 310 nM T97136 C6O0GM 145972396 IC50 = 700 nM T97136 CGN0E7 145972578 IC50 = 1300 nM T97136 C6NJ1Q 145976485 IC50 = 9500 nM T97136 CT4B8J 145977060 IC50 = 294 nM T97136 CE6R8H 145978647 IC50 = 3350 nM T97136 C9ME3Z 152452753 IC50 = 22000 nM T97136 C1SPV6 154726271 IC50 = 33 nM T97136 C4Q5US 155511270 IC50 = 2160 nM T97136 CLGS23 155512112 IC50 = 2020 nM T97136 C0JSQ1 155513638 IC50 = 1650 nM T97136 CZUP45 155514353 IC50 = 60 nM T97136 C86ZGU 155515431 IC50 = 1500 nM T97136 C09XWD 155516400 IC50 = 1080 nM T97136 C3FH8B 155516612 IC50 = 120 nM T97136 CY4J6T 155518079 IC50 = 1880 nM T97136 CK0Q8W 155518399 IC50 = 1390 nM T97136 C1HKU4 155518946 IC50 = 1700 nM T97136 CQ4W1E 155519145 IC50 = 1000 nM T97136 CBQ3S2 155519738 IC50 = 1220 nM T97136 C2QJ5U 155520323 IC50 = 1260 nM T97136 CZB7S9 155520845 Ki = 32 nM T97136 CQFN95 155520992 IC50 = 940 nM T97136 CF19DM 155521087 IC50 = 880 nM T97136 C8J4WF 155521346 IC50 = 930 nM T97136 C7MWN9 155522650 IC50 = 1680 nM T97136 CKR24E 155522757 IC50 = 1820 nM T97136 C2P7HQ 155522861 IC50 = 3700 nM T97136 CO5T8P 155523016 IC50 = 12000 nM T97136 C9C2LP 155523401 IC50 = 2220 nM T97136 CL9KF7 155523960 Ki = 221 nM T97136 C9P5BJ 155525376 IC50 = 1500 nM T97136 C5GD1C 155525441 IC50 = 1470 nM T97136 CT6PH0 155526131 IC50 = 400 nM T97136 C3EL4A 155526234 IC50 = 11000 nM T97136 CTB5M2 155526676 IC50 = 1990 nM T97136 C8TP3D 155527086 IC50 = 1150 nM T97136 CC58XT 155527888 IC50 = 1690 nM T97136 C6DVW8 155528856 IC50 = 130 nM T97136 CK3PQ6 155529232 IC50 = 2110 nM T97136 C4AY9Z 155529403 IC50 = 650 nM T97136 C58NSR 155530181 IC50 = 1500 nM T97136 CV94BT 155530828 IC50 = 2040 nM T97136 CTY27J 155531123 IC50 = 2020 nM T97136 CBJ71H 155531160 IC50 = 900 nM T97136 CIO69B 155532028 Ki = 341 nM T97136 CMX02J 155532207 IC50 = 1100 nM T97136 CY92RD 155532679 IC50 = 1100 nM T97136 CA6XT4 155533012 IC50 = 2140 nM T97136 CX98RF 155534413 IC50 = 1400 nM T97136 C4QC5Z 155535305 IC50 = 1870 nM T97136 CHBK90 155535539 IC50 = 1120 nM T97136 CRDU56 155535663 IC50 = 2290 nM T97136 C8V7IT 155536337 IC50 = 1900 nM T97136 CF6TV0 155536764 IC50 = 1540 nM T97136 CZOW93 155537061 IC50 = 58000 nM T97136 C52MTP 155537215 IC50 = 8400 nM T97136 C8P7BM 155537933 IC50 = 1500 nM T97136 C6GHV2 155538859 IC50 = 1690 nM T97136 C3GT7O 155539850 IC50 = 1740 nM T97136 C12SQW 155540442 IC50 = 1250 nM T97136 C59FGZ 155541299 IC50 = 1100 nM T97136 C6ZOE2 155541823 IC50 = 2290 nM T97136 CY1JU6 155542746 IC50 = 930 nM T97136 CN5KT8 155544930 IC50 = 2080 nM T97136 C6XV2T 155545139 IC50 = 1810 nM T97136 C90SCP 155545296 IC50 = 2130 nM T97136 CH7LV8 155545541 IC50 = 4300 nM T97136 CSY2X6 155545770 IC50 = 14200 nM T97136 CZX2O3 155546420 IC50 = 1340 nM T97136 C47TYE 155546525 IC50 = 29300 nM T97136 C0Q8DT 155546829 IC50 = 830 nM T97136 CY07FU 155547431 IC50 = 2400 nM T97136 C1F8ET 155547855 IC50 = 1560 nM T97136 CKE71S 155548047 Ki = 76 nM T97136 CQV4G6 155548114 IC50 = 1280 nM T97136 CSM6J8 155548546 IC50 = 1000 nM T97136 C8YS9T 155548849 IC50 = 1920 nM T97136 C2OJ9K 155549245 IC50 = 820 nM T97136 C25ZXE 155549543 IC50 = 1730 nM T97136 CA1N4E 155550773 IC50 = 1090 nM T97136 CP0C5Q 155551458 IC50 = 2060 nM T97136 CQP94O 155551694 IC50 = 1070 nM T97136 CU2VF4 155553572 IC50 = 1850 nM T97136 CE4M8Y 155555762 IC50 = 8000 nM T97136 CA49YB 155555925 IC50 = 1890 nM T97136 CJ81CB 155555985 IC50 = 970 nM T97136 CWN95Z 155556129 IC50 = 1650 nM T97136 CZ5V1L 155556205 IC50 = 1570 nM T97136 C2ACZ9 155557322 IC50 = 2350 nM T97136 C94QIK 155557622 IC50 = 1100 nM T97136 CE9LF8 155558154 IC50 = 1620 nM T97136 C8QN5S 155558190 IC50 = 1720 nM T97136 CW4SI7 155558796 IC50 = 1360 nM T97136 C0YZ6T 155559185 IC50 = 1390 nM T97136 CX2JF3 155559188 IC50 = 1650 nM T97136 CB5NR2 155559630 IC50 = 2800 nM T97136 C1NVA6 155560651 IC50 = 54 nM T97136 C83AYT 155560735 IC50 = 2500 nM T97136 C89HUQ 155560889 IC50 = 1380 nM T97136 CEY5K6 155561325 IC50 = 1950 nM T97136 C7X8VA 155561466 IC50 = 1410 nM T97136 CE6Y0J 155561742 IC50 = 1900 nM T97136 C0S1RX 155562041 IC50 = 1640 nM T97136 COV53N 155562214 IC50 = 1540 nM T97136 CGF1C5 155564109 IC50 = 4400 nM T97136 C58CFL 155564724 IC50 = 2170 nM T97136 C0CGY2 155565497 IC50 = 2240 nM T97136 C86CBS 155565872 IC50 = 1460 nM T97136 C3YLD0 155565921 IC50 = 2190 nM T97136 CGH65C 155566572 IC50 = 310 nM T97136 CQ25XI 155566821 IC50 = 1900 nM T97136 C37BGO 155567311 IC50 = 200 nM T97136 CYA3E9 155567459 IC50 = 85 nM T97136 CS84WB 155567583 IC50 = 1630 nM T97136 C1LUJ4 155567803 IC50 = 1160 nM T97136 C9LM2V 155567962 IC50 = 1310 nM T97136 C4AY9W 155568101 IC50 = 2200 nM T97136 CVNW62 155569155 IC50 = 1100 nM T97136 C8AOM4 11724428 IC50 = 40000 nM T97136 C13GYL 127031746 IC50 < 5000 nM T97136 D01KOI 346926 IC50 = 57000 nM T97136 D01WIH 51998 IC50 = 1030 nM T97136 D03ATU 4707 IC50 = 1700 nM T97136 D03BJF 44465558 IC50 = 19000 nM T97136 D03DZO 11715767 IC50 = 2670 nM T97136 D0A7FQ 11644425 IC50 = 870 nM T97136 D0EW9J 10389239 IC50 = 5700 nM T97136 D0N7AJ 11409972 IC50 = 1760 nM T97136 D0W6VA 82315 IC50 = 13000 nM T97136 D0Y0BK 11524144 IC50 = 11 nM T97136 D0ZH1U 2051 IC50 = 530 nM T92424 D01TJY 53340771 IC50 = 2 nM T92424 D09ZXO 176873 IC50 = 2.1 nM T92424 C2E9ZX 3080994 IC50 = 92000 nM T92424 CY7WS4 9799158 IC50 = 43000 nM T92424 C4LTP2 9825687 IC50 = 0.77 nM T92424 CB0JO4 9826672 IC50 = 0.5 nM T92424 CQ25XG 9827352 IC50 = 2.2 nM T92424 CO16RP 9828120 IC50 = 1.4 nM T92424 CB8GP1 9828375 IC50 = 2.5 nM T92424 CJ9HV0 9828819 IC50 = 11 nM T92424 C87ADQ 9830626 IC50 = 1.7 nM T92424 CSJ1Z5 9846189 IC50 = 0.21 nM T92424 CZ0AS2 9846634 IC50 = 0.7 nM T92424 CY63LZ 9846660 IC50 = 149 nM T92424 CVXG48 9862253 IC50 = 33 nM T92424 CHC56Q 9870640 IC50 = 72 nM T92424 C5EJN9 9884317 IC50 = 2.5 nM T92424 CV4T6H 9885053 IC50 = 140 nM T92424 C6PNG8 9894403 IC50 = 540 nM T92424 CNX29T 9907082 IC50 = 23 nM T92424 CC6PJ4 9908437 Ki = 6 nM T92424 CF4J2Z 9923982 IC50 = 210 nM T92424 CUBV32 9924032 IC50 = 420 nM T92424 CJPZ87 9930471 IC50 = 0.8 nM T92424 C1UK7T 9953715 Ki = 2.5 nM T92424 C4XK2S 9956830 IC50 = 470 nM T92424 CDU79H 9957105 IC50 = 6.4 nM T92424 CT4V2Y 9979833 IC50 = 17.5 nM T92424 CXN45H 9983052 IC50 = 17 nM T92424 CA2SU9 10004734 IC50 = 1.47 nM T92424 CY0T9L 10030149 IC50 = 16 nM T92424 CE2CK1 10032445 IC50 = 546000 nM T92424 COH3U6 10052945 IC50 = 18 nM T92424 C40FMW 10069462 IC50 = 0.1 nM T92424 C3WZR0 10069974 IC50 = 0.9 nM T92424 CLN76R 10096459 IC50 = 2670 nM T92424 CS2A6F 10098382 IC50 = 3.27 nM T92424 C4GEW5 10111539 IC50 = 15.85 nM T92424 C1H4NB 10132697 IC50 = 33 nM T92424 CLBK65 10160411 IC50 = 15 nM T92424 CDL31V 10165701 IC50 = 3.7 nM T92424 CV0G1X 10181237 IC50 = 0.5 nM T92424 CP64AK 10181815 IC50 = 0.68 nM T92424 CO8D9C 10196873 IC50 = 310 nM T92424 C42BVA 10251325 IC50 = 9.4 nM T92424 CM9UQ8 10252576 IC50 = 11 nM T92424 C38UIQ 10273975 IC50 = 12.59 nM T92424 CD04QE 10279663 IC50 = 3.3 nM T92424 CR2YI9 10297636 IC50 = 2.1 nM T92424 CQ04DG 10367832 IC50 = 2.58 nM T92424 CQ4H3K 10386147 IC50 = 29 nM T92424 C8PNS3 10391689 IC50 = 1.86 nM T92424 CC0L8M 10392074 IC50 = 5170 nM T92424 CX1D5C 10411516 IC50 = 1.2 nM T92424 CR0F1T 10412890 IC50 = 5.43 nM T92424 CUHY62 10433896 IC50 = 1.7 nM T92424 CRP82B 10435346 IC50 = 2500 nM T92424 C1ME0S 10436235 IC50 = 3 nM T92424 C04HQK 10437073 IC50 = 1.03 nM T92424 C1EH5P 10439474 IC50 = 5.5 nM T92424 C6P0ZM 10458809 IC50 = 180 nM T92424 C9OM3L 10482416 IC50 = 1.84 nM T92424 C6R4MV 10678165 IC50 = 18000 nM T92424 C4XFU2 10767331 IC50 = 8700 nM T92424 C08BCF 10993678 IC50 = 42 nM T92424 CDK7W9 10994476 IC50 = 350 nM T92424 CTW0P5 11102917 IC50 = 39 nM T92424 C79OJR 11133736 IC50 = 1600 nM T92424 CZO3H7 11399588 IC50 = 330 nM T92424 C5NEM0 11546965 IC50 = 1.2 nM T92424 CFZ2O9 11613998 IC50 > 50000 nM T92424 CDV02G 11628719 IC50 = 5200 nM T92424 CGU84F 11721315 IC50 = 550 nM T92424 C2ONX6 11721442 IC50 = 245 nM T92424 CR2CL6 11842612 IC50 = 1.1 nM T92424 CF8YK0 11965389 IC50 = 0.96 nM T92424 CW7T9U 11965462 IC50 = 11 nM T92424 CDVB07 15850631 IC50 > 10000 nM T92424 CG9FV3 15850632 IC50 = 40 nM T92424 CDUW15 16088010 IC50 = 7960 nM T92424 CR6ZY3 16088011 IC50 = 14.3 nM T92424 CTGC60 16678135 IC50 = 1100 nM T92424 CU8YQ3 16756502 IC50 = 19 nM T92424 C0KW3V 16756505 IC50 = 30000 nM T92424 C04JOX 16756621 IC50 = 2700 nM T92424 C4CU7T 16756622 IC50 = 6800 nM T92424 CFH96E 16756623 IC50 = 3100 nM T92424 CB15RX 16756849 IC50 = 260 nM T92424 CM18ZN 16756955 IC50 = 2300 nM T92424 CL38IU 16756956 IC50 = 29 nM T92424 CW5P8L 16756957 IC50 = 4300 nM T92424 C0O6XT 19076730 IC50 = 69 nM T92424 C85SOV 20666970 IC50 = 102 nM T92424 C61WDP 20666971 IC50 = 144 nM T92424 CX52NV 20666990 IC50 = 40 nM T92424 CVJ8N2 20667011 IC50 = 0.38 nM T92424 CQ8ME6 20667015 IC50 = 0.76 nM T92424 C3TR2D 21191396 IC50 = 3 nM T92424 CGI19E 21191399 IC50 = 1 nM T92424 CN1Q0M 21191405 IC50 = 0.41 nM T92424 C3GK7N 21191409 IC50 = 135 nM T92424 CQJ5Z3 21191417 IC50 = 16.6 nM T92424 C7XYV3 21191470 IC50 = 0.96 nM T92424 CMS31G 22098946 IC50 = 29 nM T92424 CE5G2I 22098949 IC50 = 116 nM T92424 C94AUL 22098977 IC50 = 45 nM T92424 CHP6U7 22347519 IC50 = 4 nM T92424 CE2G6D 22347593 IC50 = 3 nM T92424 CIO36K 22347604 IC50 = 20 nM T92424 CXVB03 22594242 IC50 = 0.2 nM T92424 CDJH42 22594251 IC50 = 0.3 nM T92424 CPF73W 22594331 IC50 = 20 nM T92424 CHR03I 22594351 IC50 = 22 nM T92424 CFL7X5 22594355 IC50 = 119 nM T92424 CY6WR2 24872066 IC50 = 15000 nM T92424 CUM4E3 24872070 IC50 = 11700 nM T92424 CG09DH 24872646 IC50 = 1870 nM T92424 CRS65Q 24873110 IC50 = 11500 nM T92424 C0HZ7E 24873345 IC50 = 8290 nM T92424 CM37RS 42607047 IC50 = 2.7 nM T92424 C7K4HE 42607050 IC50 = 44 nM T92424 CF7C8I 44283067 IC50 = 3.1 nM T92424 C12RPS 44283197 IC50 = 13 nM T92424 C4VW3I 44283198 IC50 = 9.6 nM T92424 C9ZQW4 44283202 IC50 = 60 nM T92424 C6KLR5 44283203 IC50 = 39 nM T92424 C74CWT 44283235 IC50 = 8.1 nM T92424 CVS5P4 44283263 IC50 = 26 nM T92424 CX2PH8 44283275 IC50 = 49 nM T92424 C2M4JN 44283364 IC50 = 7.6 nM T92424 CNFY65 44291131 IC50 = 300 nM T92424 CUZ73G 44291499 IC50 = 10 nM T92424 C4LEU0 44340569 IC50 = 40 nM T92424 CR51ID 44378699 IC50 > 10000 nM T92424 CAO29R 44378701 IC50 = 10000 nM T92424 CWP41H 44378720 IC50 = 5800 nM T92424 C2U6ZA 44378747 IC50 = 10000 nM T92424 CT9H2B 44378748 IC50 > 10000 nM T92424 CNS75M 44378858 IC50 = 10000 nM T92424 CENU52 44378961 IC50 = 4300 nM T92424 C3UQT1 44378995 IC50 = 5820 nM T92424 CHC7N5 44379066 IC50 = 4300 nM T92424 CVYB52 44393453 IC50 > 20000 nM T92424 CS2I9D 44394317 IC50 = 1000 nM T92424 C0IN2J 44395933 IC50 = 2.2 nM T92424 CL1AJ8 44395975 IC50 = 270 nM T92424 CK4YH8 44396023 IC50 = 36 nM T92424 C3DN8C 44396062 IC50 = 8.7 nM T92424 CZ4O2D 44407529 IC50 = 2.9 nM T92424 C1E7HF 44407560 IC50 = 4.6 nM T92424 C7CP1X 44407779 IC50 = 4 nM T92424 CB5R4A 44408398 IC50 > 1000 nM T92424 C43TRL 44408407 IC50 > 1000 nM T92424 CKQ84P 44423882 IC50 = 3 nM T92424 CX1C4T 44552445 IC50 = 315 nM T92424 CT0PO4 44606192 IC50 = 114 nM T92424 C5PZ8G 46201042 IC50 = 22.95 nM T92424 C89ZFA 46224777 IC50 = 3540 nM T92424 C5X1NZ 46224858 IC50 = 12400 nM T92424 CDG6B1 46224859 IC50 = 15600 nM T92424 CKM2X1 46224860 IC50 = 32.1 nM T92424 CL39GY 46224861 IC50 = 3320 nM T92424 C56PVC 46226894 IC50 = 90700 nM T92424 CVXH79 46226896 IC50 = 1340 nM T92424 CBKZ57 46226897 IC50 = 347 nM T92424 C30JXH 46226899 IC50 = 502 nM T92424 C2WHK1 46226900 IC50 = 3569 nM T92424 C5H9YT 46226901 IC50 > 20 nM T92424 CV8W7P 46226902 IC50 = 1700 nM T92424 C83EWD 46226903 IC50 = 2475 nM T92424 CRVU54 46226904 IC50 > 2000 nM T92424 CE85AX 46226905 IC50 = 257 nM T92424 C81VUL 46229417 IC50 = 0.37 nM T92424 CNP0O2 46229418 IC50 = 9500 nM T92424 CPB51X 46229419 IC50 = 8.39 nM T92424 CC6HP8 46229421 IC50 = 6.5 nM T92424 C1CR9Y 46229422 IC50 = 59.9 nM T92424 CR53AM 46229424 IC50 = 11800 nM T92424 C81NZJ 49782807 IC50 > 10000 nM T92424 C17UYM 49782809 IC50 > 10000 nM T92424 CNT47C 49782811 IC50 > 10000 nM T92424 CK52QA 49782813 IC50 > 10000 nM T92424 CCX41K 49783020 IC50 = 1.02 nM T92424 CP7U9T 50907449 IC50 > 10000 nM T92424 C59LHA 52941929 IC50 > 10000 nM T92424 C04OYX 52942589 IC50 > 10000 nM T92424 C69YHV 52943199 IC50 = 1780 nM T92424 C8AS0O 52943382 IC50 = 2420 nM T92424 CEF0A3 52945622 IC50 = 46300 nM T92424 C7MW0D 52948102 IC50 = 1020 nM T92424 C5T8DB 52948257 IC50 > 10000 nM T92424 C5K2ME 52948941 IC50 = 1270 nM T92424 CF10XI 52949257 IC50 > 10000 nM T92424 CV9B3M 52950165 IC50 = 4380 nM T92424 C94QEJ 57521432 IC50 = 216 nM T92424 C1RDQ5 57521434 IC50 = 79 nM T92424 CT7FL5 57523172 IC50 = 149 nM T92424 C31IUF 69863577 IC50 > 10000 nM T92424 C5G9BX 71449526 IC50 = 0.76 nM T92424 C1GAT7 71451321 IC50 = 1 nM T92424 CQ0U6Z 71451322 IC50 = 0.73 nM T92424 C2TCV3 71454875 IC50 = 2.05 nM T92424 COJ71C 71454876 IC50 = 2.2 nM T92424 C5Q3PB 71461030 IC50 = 75 nM T92424 C9DS7U 71461032 IC50 > 5000 nM T92424 C8EM7Y 71550913 IC50 = 227 nM T92424 CU95LC 71574160 IC50 > 10000 nM T92424 COJ8Y4 71574161 IC50 > 10000 nM T92424 C8V4UB 71574356 IC50 > 10000 nM T92424 C8B7QE 72949858 IC50 = 61 nM T92424 CZ2P8U 73345565 IC50 = 2200 nM T92424 CQAE56 73345568 IC50 > 10000 nM T92424 CU1VZ5 73345570 IC50 = 9900 nM T92424 CPT7S8 73345576 IC50 = 7140 nM T92424 CZ6Y9R 73347081 IC50 = 4030 nM T92424 CZ35TD 73347085 IC50 = 3460 nM T92424 CGM9F7 73347087 IC50 = 10000 nM T92424 C89ENA 73347090 IC50 = 6700 nM T92424 CN1A2D 73347092 IC50 = 1580 nM T92424 CO9L2V 73348591 IC50 = 9470 nM T92424 C43LWV 73348592 IC50 = 4250 nM T92424 CM37AE 73348593 IC50 = 1700 nM T92424 CT1RG5 73348594 IC50 = 4930 nM T92424 CF1UL2 73348680 IC50 = 1300 nM T92424 CQ5D7B 73350175 IC50 = 15300 nM T92424 C20AJB 73350179 IC50 = 8400 nM T92424 C19PJE 73350181 IC50 = 4800 nM T92424 C2F3YZ 73351673 IC50 = 7200 nM T92424 CJA25I 73351674 IC50 = 2000 nM T92424 C6NCQ1 73351675 IC50 = 7700 nM T92424 C46ULG 73351676 IC50 = 7850 nM T92424 C8B6NV 73351677 IC50 = 4900 nM T92424 CIYV49 73351678 IC50 = 10000 nM T92424 C0PU3D 73351771 IC50 = 0.35 nM T92424 C20FGN 73353141 IC50 = 10000 nM T92424 CP6AJ3 73353143 IC50 = 8800 nM T92424 CUPR57 73353147 IC50 = 340 nM T92424 C83RAM 73353150 IC50 = 4700 nM T92424 CAJ27W 73354663 IC50 = 6200 nM T92424 CT4A5S 73354664 IC50 = 6900 nM T92424 C6XTP9 73354667 IC50 = 2340 nM T92424 CZ1BL4 73354668 IC50 = 790 nM T92424 C4EJK0 73356213 IC50 = 1050 nM T92424 CH8G5C 73356216 IC50 = 6600 nM T92424 CPG36Q 73356217 IC50 = 3000 nM T92424 CD1S3N 73356221 IC50 = 8850 nM T92424 CO3WF4 73356277 IC50 = 128 nM T92424 CXM8L3 75002097 IC50 = 79.43 nM T92424 C30NBD 86272865 IC50 = 125.89 nM T92424 CW8UV5 86272868 Ki = 10 nM T92424 CI07FE 90645591 IC50 = 80000 nM T92424 CLCN89 117977916 IC50 > 10000 nM T92424 CJO3B6 117978172 IC50 > 10000 nM T92424 CY1IS6 118718872 IC50 = 10000 nM T92424 C2J3VA 118721315 IC50 = 100 nM T92424 C0BT3F 118721316 IC50 = 1584.89 nM T92424 C4TNZ0 118721317 IC50 = 19.95 nM T92424 C2N6WI 118721318 IC50 = 501.19 nM T92424 CMQ94S 118721319 IC50 = 25.12 nM T92424 C5CW9O 118721320 IC50 = 50.12 nM T92424 CYL2X3 118721321 IC50 = 63.1 nM T92424 CFQA95 118721322 IC50 = 63.1 nM T92424 CWDE71 118721323 IC50 = 125.89 nM T92424 CM9J4X 118721324 IC50 = 100 nM T92424 CY13BE 118721325 IC50 = 50.12 nM T92424 C8UNZ5 118721326 IC50 = 398.11 nM T92424 CG5B9F 118721327 IC50 = 316.23 nM T92424 CMXJ63 118721328 IC50 = 501.19 nM T92424 C2OJX9 118721329 IC50 = 398.11 nM T92424 C0YG4M 118721330 IC50 = 630.96 nM T92424 C8F4DG 118721331 IC50 = 39.81 nM T92424 C2ESU9 118721332 IC50 = 39.81 nM T92424 C2OYU9 118721333 IC50 = 63.1 nM T92424 CX0R3H 118721334 IC50 = 1995.26 nM T92424 CP8I3D 118721335 IC50 = 79.43 nM T92424 CGM28Y 118721336 IC50 = 501.19 nM T92424 COM73D 118721337 IC50 = 100 nM T92424 CH25GR 118721338 IC50 = 199.53 nM T92424 CE7D1S 118721339 IC50 = 63.1 nM T92424 CZ95CL 118721340 IC50 = 79.43 nM T92424 C0AL1C 118721341 IC50 = 398.11 nM T92424 CAZ6U3 118721342 IC50 = 63.1 nM T92424 C65KQW 118721343 IC50 = 63.1 nM T92424 CGJ9O5 118978102 IC50 = 50.12 nM T92424 CL2ER8 121242162 IC50 = 79.43 nM T92424 CPS9N3 121245322 IC50 = 199.53 nM T92424 C8P7OW 121245346 IC50 = 1995.26 nM T92424 CJ83VH 121245350 IC50 = 10000 nM T92424 CFOM46 121246727 IC50 = 100 nM T92424 CL5Q9G 121246911 IC50 = 19.95 nM T92424 CAL43C 121246982 IC50 = 50.12 nM T92424 C6XK2Y 121247103 IC50 = 6.31 nM T92424 CRG07Q 124155531 IC50 = 200 nM T92424 C69XPN 124163720 IC50 > 10000 nM T92424 C4R3BT 124163838 IC50 = 1600 nM T92424 CS2QR4 124163840 IC50 = 160 nM T92424 CR5X1T 130453989 IC50 = 19.95 nM T92424 CVT2U3 130454024 IC50 = 12.59 nM T92424 CT4BY6 130454058 IC50 = 5.012 nM T92424 CZK41V 130454091 IC50 = 25.12 nM T92424 C2OJ3C 130454093 IC50 = 39.81 nM T92424 CU73IM 131985420 IC50 = 19.95 nM T92424 CQEK82 131985476 IC50 = 39.81 nM T92424 C20ZAT 131985489 IC50 = 31.62 nM T92424 C1IKD6 131985494 IC50 = 15.85 nM T92424 CI6W9O 131985523 IC50 = 63.1 nM T92424 C57BQS 132561360 IC50 = 2511.89 nM T92424 CXZ16C 137480037 IC50 = 79.43 nM T92424 CIL96B 137632126 IC50 = 25000 nM T92424 C1CPO0 137632555 IC50 = 380000 nM T92424 CMOI37 137641477 IC50 = 2945000 nM T92424 CYS13G 137648507 IC50 = 1733000 nM T92424 CDO0Q6 137650356 IC50 = 522000 nM T92424 C4GO5B 137661340 IC50 = 26000 nM T92424 CV6JY5 139030528 IC50 = 501.19 nM T92424 CX0P5N 145982847 IC50 = 25.12 nM T92424 CL13NC 145982905 IC50 = 19.95 nM T92424 C4N5TW 145983050 IC50 = 158.49 nM T92424 CJ70YV 145984499 IC50 = 7.943 nM T92424 C4R5NQ 145984560 IC50 = 199.53 nM T92424 CM9FS1 145985439 IC50 = 251.19 nM T92424 CRA6D0 145985939 IC50 = 3.162 nM T92424 CHT1J6 155515540 IC50 > 1000 nM T92424 CQ5C4M 155516533 IC50 > 1000 nM T92424 C35OHK 155518750 IC50 = 158.49 nM T92424 CTA5S4 155518784 IC50 = 251.19 nM T92424 CJ7O2X 155534687 IC50 > 1000 nM T92424 CR36QP 155540115 IC50 > 10000 nM T92424 CWF98D 155552156 IC50 > 1000 nM T92424 CKRE58 155563328 IC50 = 1000 nM T92424 CEF3T8 155563936 IC50 > 1000 nM T92424 C1HNT9 155567705 IC50 = 79.43 nM T92424 C7Z4RD 155569291 IC50 = 630.96 nM T92424 D00YBU 10699123 IC50 = 15.65 nM T92424 D01BZH 11613122 IC50 = 125.4 nM T92424 D01MGI 11583738 IC50 = 0.59 nM T92424 D03KLT 24822283 IC50 = 86.6 nM T92424 D03YLY 24822953 IC50 = 30 nM T92424 D04WVG 11540460 IC50 = 13.1 nM T92424 D05EWB 10416726 IC50 = 3.4 nM T92424 D05GXK 24822444 IC50 = 89.2 nM T92424 D05VEC 11712622 IC50 = 6.56 nM T92424 D06JLN 11518823 IC50 = 4.56 nM T92424 D06LUT 44379110 IC50 = 5270 nM T92424 D07QJD 24822784 IC50 = 1.87 nM T92424 D07UOF 44408450 IC50 = 19.81 nM T92424 D07WDB 104802 IC50 = 38000 nM T92424 D08CFM 11505585 IC50 = 42.8 nM T92424 D09PLA 11533023 IC50 = 3.43 nM T92424 D0A0KS 9851104 IC50 = 0.11 nM T92424 D0H4EK 11643340 IC50 = 93.9 nM T92424 D0J6SP 24824620 IC50 = 154 nM T92424 D0LF7W 11569720 IC50 = 411.5 nM T92424 D0M0BN 11636164 IC50 = 93.5 nM T92424 D0M6NQ 10372586 IC50 = 7.7 nM T92424 D0O6DN 11584047 IC50 = 29.6 nM T92424 D0O9FL 24823110 IC50 = 36.1 nM T92424 D0R3CY 9952958 Ki = 1.3 nM T92424 D0R9GW 11540715 IC50 = 165.5 nM T92424 D0R9SJ 44439175 IC50 = 0.9 nM T92424 D0U2NV 44408397 IC50 = 72.7 nM T92424 D0UE7H 11670104 IC50 = 26 nM T92424 D0V0JC 9986643 IC50 = 10.03 nM T92424 D0W6CJ 11656381 IC50 = 1300 nM T92424 D0Z6WZ 24822282 IC50 = 94 nM T00043 D07POC 176870 IC50 = 910 nM T00043 D09XZB 123631 IC50 = 420 nM T00043 D0F8DL 176155 IC50 = 105 nM T00043 D0Q7HO 4705 IC50 = 260 nM T00043 C7YRI8 5328840 IC50 = 130 nM T00043 CC2E4Q 5330468 IC50 = 2.4 nM T00043 C1YWE0 5330475 IC50 = 23 nM T00043 C3ZC6E 16045442 IC50 = 72 nM T00043 CHOK82 25000333 IC50 = 500 nM T00043 CU58ZC 44331212 IC50 = 510 nM T00043 CI3JR0 44532526 IC50 = 170 nM T00043 C3VRO9 44557921 IC50 > 10000 nM T00043 C67OJG 44588117 Ki = 1750 nM T00043 CK9Y2G 46197129 IC50 = 4200 nM T00043 CZC9M5 67469084 Ki = 220 nM T00043 CH29GF 71258526 IC50 > 10 nM T00043 CCNF57 132019696 Ki = 49 nM T00043 C4YWO9 134812845 Ki = 1700 nM T00043 CG15PY 134812846 Ki = 3.1 nM T00043 CGB0R3 135567262 IC50 = 0.06 nM T00043 C9O8CQ 137348448 Ki = 1600 nM T00043 C63TGO 137349551 Ki = 870 nM T00043 C6I5ME 137349552 Ki = 2600 nM T00043 CRC8D2 155489850 Ki = 2500 nM T00043 CD46IN 155514865 IC50 = 31 nM T00043 CG8J5X 155518911 Ki = 510 nM T00043 CQFC65 155533189 IC50 = 2600 nM T00043 CAN08J 155534113 Ki = 360 nM T00043 C16JRL 155535406 Ki = 3200 nM T00043 C3XR8O 155536206 Ki = 4600 nM T00043 CX68YN 155541385 Ki = 19000 nM T00043 CWU67H 155543077 Ki = 3900 nM T00043 CD8K3O 155543384 Ki = 780 nM T00043 CUTW39 155546618 Ki = 1700 nM T00043 C4E0HB 155546757 Ki = 7000 nM T00043 C49UVQ 155547733 Ki = 2900 nM T00043 CI2J4O 155551330 Ki = 3200 nM T00043 CP2K8O 155554487 Ki = 1100 nM T00043 CS8MC1 155562025 Ki = 580 nM T00043 C8UW4P 155562878 Ki = 1300 nM T00043 CDP94M 155569521 Ki = 4600 nM T00043 D0L4HJ 5330462 IC50 = 350 nM T60003 D0K8KX 5280343 IC50 = 5800 nM T60003 D03KKR 3547 IC50 = 1700 nM T60003 D03LWG 53235510 IC50 > 10000 nM T60003 D07EHV 44814409 IC50 = 4900 nM T60003 D0E3TC 44259 IC50 = 1 nM T60003 C8IAR2 5281657 IC50 = 54900 nM T60003 CI68PW 5283685 IC50 > 100000 nM T60003 CXK0S6 5283727 IC50 > 100000 nM T60003 C4G9WR 9547398 IC50 > 100000 nM T60003 C76CUP 9547698 IC50 > 100000 nM T60003 CR8DA1 10024683 IC50 > 100000 nM T60003 CLA93G 10047202 IC50 > 100000 nM T60003 C3LCH5 10047545 IC50 > 100000 nM T60003 C4CP7K 10423452 IC50 = 45300 nM T60003 C83QWV 10714343 IC50 > 100000 nM T60003 C8G5WP 11210533 IC50 = 9000 nM T60003 C7YG1N 24759534 IC50 = 3900 nM T60003 C1ONA4 24996161 IC50 = 35 nM T60003 C3VRO9 44557921 IC50 > 10000 nM T60003 CSV5B9 46901859 IC50 = 7 nM T60003 C2W9OA 53324451 IC50 > 10000 nM T60003 C1XS2J 54760383 IC50 = 6100 nM T60003 C9ZFS1 54764923 IC50 > 100000 nM T60003 CXJ63M 59603829 IC50 = 18000 nM T60003 CQEU96 59603842 IC50 = 250 nM T60003 C1HSE0 67035086 IC50 = 2600 nM T60003 CWI6K5 67035106 IC50 = 9700 nM T60003 CV63UL 67240318 IC50 > 10000 nM T60003 C8I7GC 68293638 IC50 > 10000 nM T60003 CD56XK 68293660 IC50 > 10000 nM T60003 C5DGR9 69036886 IC50 = 10000 nM T60003 C0DL3F 72698602 IC50 < 1 nM T60003 C3UC9H 73891099 IC50 = 4480 nM T60003 CV8QX0 76310169 IC50 > 30000 nM T60003 CA5L4W 76324771 IC50 > 30000 nM T60003 C9GO0P 76328313 IC50 = 18600 nM T60003 C39FTZ 76335685 IC50 > 100000 nM T60003 CSV23A 78673872 IC50 = 547 nM T60003 CPG3A5 86302574 IC50 > 30000 nM T60003 C1HW4B 89735655 IC50 = 17000 nM T60003 CN67RP 91758287 IC50 > 1000 nM T60003 C7ZL3Q 118715599 IC50 = 99 nM T60003 C8T0AY 118715600 IC50 = 990 nM T60003 C2J3YZ 118715601 IC50 > 1000 nM T60003 CRG06J 118715602 IC50 > 1000 nM T60003 C7WS3V 118715603 IC50 > 1000 nM T60003 CQM81J 118715604 IC50 > 1000 nM T60003 C2MD1Q 155513187 IC50 > 10000 nM T60003 D06HVH 54613583 IC50 = 310 nM T00216 D01AZG 5073 Ki = 0.69 nM T00216 D01UXC 2249 IC50 = 230 nM T00216 D03SKR 2803 EC50 = 290 nM T00216 D05DVP 5717 IC50 > 10000 nM T00216 D06XZR 27400 Ki = 75 nM T00216 D07MOX 439260 Ki = 2600 nM T00216 D0AE3X 2435 Ki = 1800 nM T00216 D0D1AL 3559 Ki = 5.7 nM T00216 D0E9PK 4810 Ki > 30000 nM T00216 D0H7KF 5002 Ki = 4.5 nM T00216 D0I8FI 3779 EC50 = 1.5 nM T00216 D0MT0M 2216 EC50 = 180 nM T00216 D0R1JV 60854 Ki = 1.9 nM T00216 D0R6BI 3341 Ki = 151.36 nM T00216 D0T6QX 5736 Ki = 3.4 nM T00216 D0T7OW 681 Ki = 2511.89 nM T00216 D0V4QS 135398745 Ki = 7.3 nM T00216 D0WV3U 4893 Ki = 0.054 nM T00216 D0X6BV 6918314 IC50 = 1980 nM T00216 D0Z1RV 135398737 Ki = 3.7 nM T00216 D07WHS 5312115 EC50 > 1000000 nM T00216 D0F2ML 68602 EC50 = 1165 nM T00216 D07YLK 4350931 Ki = 11 nM T00216 D01WJZ 60820 Ki = 1.3 nM T00216 D02FNU 56971 IC50 = 500 nM T00216 D06DZI 107780 Ki < 1000 nM T00216 D08SOF 5405 IC50 = 2340 nM T00216 D0BC6Q 9837551 Ki = 470 nM T00216 D0EE6L 3038495 Ki = 5 nM T00216 D0K0DB 6604887 Ki = 180 nM T00216 D0K9JP 9928332 Ki > 1000 nM T00216 D0O9EM 208928 Ki > 10000 nM T00216 D0OS6O 60149 Ki = 1.8 nM T00216 D0W7IR 9887884 Ki = 3900 nM T00216 D0Y1PG 9841972 EC50 = 5600 nM T00216 D0ZG9N 132337 Ki > 10000 nM T00216 C4JQ7T 2068 Ki > 100000 nM T00216 CZUI83 2769 IC50 = 30 nM T00216 CK1JY9 3106 Ki = 1995.26 nM T00216 C0H8GR 3191 IC50 = 183 nM T00216 C2H1VA 131829 Ki = 1100 nM T00216 CZL87W 133999 IC50 > 10000 nM T00216 CF4V5Q 185076 Ki = 1400 nM T00216 C64CQL 385013 Ki = 76 nM T00216 C1VE3T 386224 Ki = 79 nM T00216 CT3UV7 444005 IC50 > 1000 nM T00216 CJ30IQ 1248739 Ki = 260 nM T00216 C64CZV 3038494 Ki = 5 nM T00216 C54QJC 3086247 Ki = 2400 nM T00216 CWNZ35 6469693 Ki = 98 nM T00216 CJTQ40 6469918 Ki = 60 nM T00216 C9R7NM 9104271 IC50 = 88 nM T00216 CHD32K 9794524 Ki > 28000 nM T00216 C4K7ZJ 9795515 Ki = 4200 nM T00216 CLUT03 9799123 IC50 = 1257 nM T00216 CCSN93 9800737 IC50 = 1000 nM T00216 CX7I8J 9802187 Ki = 16 nM T00216 CX3U7N 9813501 Ki = 430 nM T00216 CJM0W8 9816863 Ki = 2300 nM T00216 C45QPU 9820163 Ki = 1 nM T00216 C95BXW 9823464 IC50 = 100 nM T00216 CJ8LT7 9848518 IC50 > 10000 nM T00216 CB31LS 9855978 Ki = 1200 nM T00216 CTUM52 9856417 Ki = 1700 nM T00216 C3YSQ5 9859238 Ki = 5100 nM T00216 CQ2L0J 9859437 Ki = 16000 nM T00216 C7EZ2L 9859861 Ki > 10000 nM T00216 C5WYN4 9865858 Ki = 53 nM T00216 C3GMU5 9868889 Ki = 1.2 nM T00216 CA87LO 9869262 Ki = 56.23 nM T00216 CT2C6K 9870702 IC50 > 10000 nM T00216 CK76MQ 9872238 Ki = 0.4 nM T00216 CYSB08 9878065 Ki = 730 nM T00216 CPI8G9 9881158 Ki = 1500 nM T00216 C3DB5H 9884781 Ki = 967 nM T00216 C9GB2M 9888555 Ki = 15 nM T00216 CDLB96 9889149 IC50 = 100 nM T00216 C1ANB8 9889726 Ki = 1.99 nM T00216 C6CZ3G 9906777 IC50 > 10000 nM T00216 CO7BK6 9909648 Ki = 38 nM T00216 CQ3L1X 9921302 Ki = 670 nM T00216 CJ46NU 9921303 Ki = 490 nM T00216 CBE1Y9 9921863 Ki = 3300 nM T00216 CH5D3J 9928343 IC50 > 10000 nM T00216 C5V0UE 9933975 Ki = 41.1 nM T00216 C5E7KC 9943680 Ki = 3200 nM T00216 C1K8WB 9951233 Ki = 2003 nM T00216 C4I7UJ 9964754 Ki = 1000 nM T00216 CQIU94 9978693 IC50 = 700 nM T00216 CC6M7Z 9980998 Ki > 10000 nM T00216 C2C1XS 10042602 Ki = 67.61 nM T00216 C2JZL1 10048222 IC50 > 1000 nM T00216 C4GHO2 10053476 Ki > 1000 nM T00216 CJXQ40 10092819 Ki = 8.6 nM T00216 CRS5B6 10176999 Ki = 2100 nM T00216 CQ8HX2 10198135 Ki = 8400 nM T00216 C6S2RA 10198552 Ki = 130 nM T00216 CC2KV3 10214826 Ki > 100000 nM T00216 CE9Y8J 10276451 Ki = 370 nM T00216 C9LWG3 10369004 IC50 = 59 nM T00216 CS2DN8 10376336 EC50 = 12692 nM T00216 C69KIB 10385855 IC50 > 10000 nM T00216 C4UN0A 10436653 Ki = 15 nM T00216 C8KD1B 10438027 Ki = 300 nM T00216 CO7IV6 10450593 Ki = 8 nM T00216 CIA16B 10457445 Ki = 389.05 nM T00216 C26KCR 10475231 Ki = 100 nM T00216 CPI5M7 10476504 Ki = 26 nM T00216 C48BRW 10546334 Ki = 93.33 nM T00216 CBOS60 10548781 Ki = 38 nM T00216 C6O9CB 10572092 Ki > 500 nM T00216 C1DXO0 10609673 Ki = 6600 nM T00216 CFC42Z 10664759 Ki = 47 nM T00216 CI0GO3 10666853 Ki = 234 nM T00216 CTSY18 10682720 Ki = 16000 nM T00216 C3LDA1 10690393 Ki = 44 nM T00216 CP0B6F 10691211 Ki = 33 nM T00216 CYRG83 10714368 Ki = 94 nM T00216 C0USP7 10718592 Ki = 1.7 nM T00216 C3OCI1 10731942 Ki = 16 nM T00216 C4EZS5 10736855 Ki = 132 nM T00216 C5Z3JE 10737897 Ki = 2.3 nM T00216 CIZ05K 10761543 Ki = 74 nM T00216 C9HWI2 10783359 Ki = 18 nM T00216 CG12BP 10784327 Ki > 500 nM T00216 C3P2VZ 10785265 Ki = 23 nM T00216 C1P4GW 10785266 Ki = 20 nM T00216 C81PIH 10807090 Ki = 117 nM T00216 CD92GV 10832838 Ki = 35 nM T00216 C9A8KN 10862425 Ki = 19 nM T00216 CMV36C 10884046 Ki = 48 nM T00216 CRI50E 10885636 IC50 = 1100 nM T00216 CX65PW 10907460 IC50 = 993 nM T00216 CU09AV 10937901 IC50 = 1330 nM T00216 CSLT97 10949380 IC50 = 4920 nM T00216 C2HP7F 10981761 IC50 = 4250 nM T00216 CJC9K4 11005810 IC50 = 417 nM T00216 CB7N1P 11035765 IC50 = 174 nM T00216 CFJG64 11059058 IC50 = 1340 nM T00216 CG41BK 11071079 IC50 = 1640 nM T00216 C7DE0U 11113605 IC50 = 1170 nM T00216 C75WKP 11176199 IC50 = 45 nM T00216 C8JW3Z 11260311 Ki = 140 nM T00216 C4S2VF 11277147 Ki > 1000 nM T00216 CJS9C0 11304851 IC50 = 1000 nM T00216 CN63TR 11504230 Ki = 2.5 nM T00216 C16TWK 11508052 IC50 > 10000 nM T00216 C59SCV 11516033 Ki = 61 nM T00216 CW68BJ 11518143 IC50 = 1000 nM T00216 CXWO08 11522273 IC50 > 10000 nM T00216 CY5I0U 11559581 Ki = 380 nM T00216 CNH1K4 11568826 Ki = 13.7 nM T00216 C8CU1X 11581237 Ki = 64 nM T00216 C4L7TV 11662592 Ki = 118.1 nM T00216 CTK8R9 11678172 Ki = 80 nM T00216 CEQ6W7 11694810 Ki > 1000 nM T00216 C1W8NR 11696910 Ki = 190 nM T00216 CKT7L2 11698732 Ki = 2.64 nM T00216 CB4H2O 11699469 Ki = 8.4 nM T00216 CJL61W 11706497 Ki = 480 nM T00216 CGO56C 11720302 Ki = 45 nM T00216 C7PVL8 11730467 IC50 = 2190 nM T00216 CPG15O 11743399 IC50 > 1000 nM T00216 C2J7KO 11751611 Ki = 17.26 nM T00216 CW0UA2 11792453 Ki = 348 nM T00216 CN9M8E 11811722 IC50 = 2830 nM T00216 CN9H3J 11820372 EC50 = 2113 nM T00216 C8EDN0 12088080 Ki = 300 nM T00216 C8RB6W 12088082 Ki > 1000 nM T00216 CRN3S9 13387299 Ki = 9800 nM T00216 CPA2O9 13387301 Ki = 1160 nM T00216 CIDB37 13387304 Ki = 10300 nM T00216 CXS0R8 13387308 Ki = 99000 nM T00216 C1LXY9 13473217 Ki = 6900 nM T00216 C9BQ5D 13473220 Ki = 2000 nM T00216 CLYK03 13538579 Ki = 2250 nM T00216 CES6X1 13538583 Ki = 7400 nM T00216 C36HGR 13538585 Ki = 26000 nM T00216 CV6FD5 13720763 Ki = 1970 nM T00216 CI21BN 14934406 Ki = 17 nM T00216 CAF40B 15181802 IC50 = 8 nM T00216 C2XUE8 15344574 Ki = 36 nM T00216 CEOS76 15523910 Ki = 5915 nM T00216 C6US3O 15711850 Ki > 30000 nM T00216 C5PO3N 15711869 Ki = 1820 nM T00216 CX96HP 18411849 IC50 > 1000 nM T00216 COA7W4 19079030 Ki = 12 nM T00216 CT7XG9 21830793 Ki = 6.75 nM T00216 CYH4J9 22002244 Ki = 0.1 nM T00216 C5SI3U 22464564 Ki = 6780 nM T00216 CJ6WF3 22464606 Ki = 14.8 nM T00216 CA5BY9 22464614 Ki = 8.4 nM T00216 CQB94R 22464634 Ki = 121.1 nM T00216 CAZ23L 22464649 Ki = 13.2 nM T00216 CJCY98 22464720 Ki = 1 nM T00216 CB97XC 22464804 Ki = 4.5 nM T00216 C9MB7K 22464806 Ki = 0.1 nM T00216 C7DXE6 22464831 Ki = 1.7 nM T00216 C76FEA 22464842 Ki = 1.8 nM T00216 C0I2HU 24769156 Ki = 50 nM T00216 C6L7KS 24887518 Ki = 1819.7 nM T00216 C7I9YB 44189144 IC50 = 430 nM T00216 CXR6K7 44212701 Ki > 1000 nM T00216 C8ORL9 44212702 Ki = 2.9 nM T00216 CN71EI 44212703 Ki = 200 nM T00216 C1FRU8 44288600 IC50 > 10000 nM T00216 C7AJ3B 44293793 Ki = 10000 nM T00216 CYUA79 44293794 Ki = 30000 nM T00216 CFDV86 44307552 Ki > 10000 nM T00216 CQRK31 44309145 Ki = 24.4 nM T00216 CHYZ41 44309146 Ki = 91.5 nM T00216 CU2Z3N 44309182 Ki = 2439 nM T00216 CMJV60 44309200 Ki = 5610 nM T00216 C8UR6M 44309202 Ki = 4512 nM T00216 CK26BL 44309367 Ki = 305 nM T00216 C8Y5ZU 44309368 Ki = 610 nM T00216 CHC12P 44309385 Ki = 305 nM T00216 CM02RX 44316058 Ki = 575.44 nM T00216 C9V1IL 44316331 Ki = 389.05 nM T00216 CW16JD 44324737 Ki > 1000 nM T00216 CA84SN 44324765 Ki > 1000 nM T00216 COA3H4 44324800 Ki = 380 nM T00216 CY04JW 44324972 Ki > 1000 nM T00216 C7OW8Y 44336061 Ki = 1118 nM T00216 C4R6LP 44341301 Ki = 23 nM T00216 CD9ZS8 44342270 IC50 = 1150 nM T00216 CJ80OW 44360984 Ki = 28 nM T00216 CS8K1A 44360992 Ki = 18 nM T00216 C3NZ7B 44361021 Ki = 32 nM T00216 CG85AM 44380820 Ki = 730 nM T00216 CT8Y5A 44393007 Ki = 379 nM T00216 CG9S1O 44393045 Ki = 200 nM T00216 CO6EY0 44393113 Ki > 1000 nM T00216 CE03ZW 44393134 Ki = 57 nM T00216 CG5UE1 44393169 Ki = 14 nM T00216 CK85EB 44393193 Ki = 27 nM T00216 CEO2W9 44393372 Ki = 5.8 nM T00216 CXP4Q7 44393393 Ki = 42 nM T00216 C6BZS0 44393403 Ki = 5.9 nM T00216 C86NED 44393411 Ki = 49 nM T00216 C9THO4 44393415 Ki = 1.7 nM T00216 C0E5HY 44400500 Ki = 5.1 nM T00216 CO8EU5 44400519 Ki = 26 nM T00216 CRX12E 44400553 Ki = 35 nM T00216 CIU18E 44400585 Ki = 5.5 nM T00216 CV8K2W 44400594 Ki = 26 nM T00216 C84RNU 44400626 Ki = 73 nM T00216 CY94SF 44400674 Ki = 9.7 nM T00216 CQ4U2P 44403210 Ki = 7.4 nM T00216 CKE6T4 44403213 Ki = 17 nM T00216 CAJX39 44403214 Ki = 12 nM T00216 C61CNS 44403219 Ki = 16 nM T00216 C5AE9L 44403220 Ki = 5.8 nM T00216 CC6XM4 44403224 Ki = 13 nM T00216 C6JB4M 44403225 Ki = 3.9 nM T00216 CGE52H 44403232 Ki = 14 nM T00216 C7W3BP 44405573 Ki = 1.1 nM T00216 CV9IR7 44405574 Ki = 0.5 nM T00216 CFG72V 44405575 Ki = 4 nM T00216 C8WSZ2 44405586 Ki = 0.1 nM T00216 CEJ0C3 44405587 Ki = 0.2 nM T00216 C4DK0U 44405655 Ki = 12.1 nM T00216 C28WCH 44405665 Ki = 18 nM T00216 CS7ZD5 44405666 Ki = 0.2 nM T00216 CIH9J0 44405669 Ki = 0.5 nM T00216 CVZO38 44405677 Ki = 0.5 nM T00216 CMK32Z 44405701 Ki = 26.7 nM T00216 CZK5L6 44405702 Ki = 129.1 nM T00216 CO7G3W 44405725 Ki = 7 nM T00216 CU1VL9 44405726 Ki = 0.2 nM T00216 CO1P3W 44405730 Ki = 1.2 nM T00216 C65PBE 44405930 Ki = 5.47 nM T00216 CBGH16 44405935 Ki = 1.63 nM T00216 CF4S3Y 44405965 Ki = 4.71 nM T00216 CT3Z8U 44405980 Ki = 3.32 nM T00216 CQ7RI8 44405981 Ki = 2.18 nM T00216 C0BI5F 44405985 Ki = 6.28 nM T00216 C1FZE7 44405991 Ki = 1.19 nM T00216 C4NC8M 44405995 Ki = 2.8 nM T00216 CVM1Y5 44406002 Ki = 4.97 nM T00216 C0R5VL 44406003 Ki = 11.71 nM T00216 C90NQJ 44406012 Ki = 4.08 nM T00216 CL5C9T 44406077 Ki = 16.4 nM T00216 C0EXA1 44407083 IC50 > 10000 nM T00216 CG87PW 44409290 Ki > 1000 nM T00216 C2HL9K 44460958 IC50 > 1000 nM T00216 CY8G5Q 44460979 IC50 > 1000 nM T00216 C8T6WQ 46888928 Ki = 2 nM T00216 C18KHC 46888985 Ki = 2 nM T00216 CK40FT 46888986 Ki = 91 nM T00216 CTJ1P2 46889013 Ki = 354 nM T00216 COPQ75 46889014 Ki = 8 nM T00216 CAM45V 46889015 Ki = 46 nM T00216 CZ3FI5 46889016 Ki > 3300 nM T00216 C4B6ZE 46889041 Ki = 1100 nM T00216 C95ZWE 54581386 IC50 > 10000 nM T00216 C2WX4J 54587281 IC50 = 4800 nM T00216 CJZ81X 71293954 Ki = 280 nM T00216 CZ35EN 71294092 Ki = 1.8 nM T00216 CDI84E 71450922 IC50 > 10000 nM T00216 C7W4RH 72734860 Ki = 790 nM T00216 C9T3LW 89638708 Ki = 64 nM T00216 CZDE01 118713090 Ki > 10000 nM T00216 C1KR9C 118713091 Ki = 350 nM T00216 CI5U1R 118713092 Ki = 450 nM T00216 C4S7WD 118713093 Ki = 1.8 nM T00216 CB8Q2E 118713094 Ki = 7.3 nM T00216 C5LFW4 118717221 Ki > 1000 nM T00216 C5OKG2 118727894 Ki = 74.13 nM T00216 CMGB38 118727895 Ki = 89.13 nM T00216 CBHT01 122377930 Ki = 979 nM T00216 CIHZ54 127025242 Ki = 250 nM T00216 CCY7P3 127025243 Ki = 339 nM T00216 CTYP30 127026133 Ki = 742 nM T00216 CX6EI2 127026750 Ki = 1525 nM T00216 C5OU1T 135409492 Ki = 266 nM T00216 C4PM9W 135515431 Ki = 12 nM T00216 CCGZ20 155530937 Ki > 10000 nM T00216 CVBC47 155535120 Ki = 1800 nM T00216 CP9TR0 10324985 Ki = 32.2 nM T00216 D01NOZ 16665072 IC50 = 27000 nM T00216 D02TQC 14928441 Ki = 17000 nM T00216 D04PBA 10015867 Ki > 1000 nM T00216 D05KUM 135446209 Ki = 80 nM T00216 D06HHJ 10490084 Ki = 11000 nM T00216 D09PIF 142067 Ki = 2500 nM T00216 D0A6GK 10489502 Ki = 6000 nM T00216 D0FU5E 10220053 Ki > 1000 nM T00216 D0G2CP 10404144 Ki = 240 nM T00216 D0L6JS 9816048 EC50 = 790 nM T00216 D0N7UE 10198248 Ki = 11000 nM T00216 D0O4BC 11776546 Ki = 5291 nM T00216 D0P5PW 132111 EC50 = 5793 nM T00216 D0S4VR 10655607 Ki = 24000 nM T00216 D0ZC4S 10632290 Ki > 100000 nM T95878 D0E3TC 44259 IC50 = 0.159 nM T95878 D03BNU 59604787 IC50 > 10000 nM T95878 C1MR8Q 60097495 IC50 > 1000 nM T95878 CV63UL 67240318 IC50 > 10000 nM T95878 CWS5C4 129245211 IC50 = 2360 nM T95878 CH91ON 129245363 IC50 = 528 nM T95878 CA2N5C 129245517 IC50 = 8850 nM T95878 C0E2RU 129245526 IC50 = 8910 nM T95878 C52PNC 129245623 IC50 = 1060 nM T95878 CEYK58 129245795 IC50 = 4120 nM T95878 CQJK71 129246093 IC50 = 170 nM T95878 C0GC7N 129246130 IC50 = 11200 nM T95878 CCF8W2 129261617 IC50 = 177 nM T95878 CG5O2J 129261641 IC50 = 434 nM T95878 C8KJ9Z 137479135 IC50 = 6110 nM T95878 CVHF30 137479140 IC50 = 2830 nM T95878 CM3A8O 139030333 IC50 = 14000 nM T95878 CM07EU 145714274 IC50 = 3220 nM T95878 C9ISH6 145925685 IC50 = 276 nM T95878 C7CH9V 146014951 IC50 = 7 nM T95878 CJB1R5 155511461 IC50 = 325 nM T95878 C2MD1Q 155513187 IC50 > 10000 nM T95878 CZ0WO7 155523990 IC50 = 1260 nM T95878 CHD09S 155543566 IC50 = 192 nM T95878 CC9LQ2 155546287 IC50 > 20000 nM T95878 D09PTP 57325421 IC50 = 19 nM T13484 CN8XM2 5311263 EC50 = 970 nM T13484 CLS96Y 6419701 EC50 = 930 nM T13484 COZF72 10322404 EC50 = 79 nM T13484 C7QRT8 11648176 EC50 = 38.9 nM T13484 CV86RF 44368508 EC50 = 58 nM T13484 CET63X 46223906 EC50 = 85.11 nM T13484 C57TYK 71569053 EC50 = 66 nM T13484 CSN3I7 71569056 EC50 = 75.86 nM T13484 CPT5S2 71718248 EC50 = 77.62 nM T13484 CKC4U7 71719457 EC50 = 104.71 nM T13484 C5P1CQ 71720690 EC50 = 89.13 nM T92057 D06XXH 11511120 IC50 = 74 nM T92057 D07POC 176870 IC50 = 1130 nM T92057 D08CDI 208908 IC50 > 1000 nM T92057 D09KTS 24821094 IC50 = 0.25 nM T92057 D09XZB 123631 IC50 = 476 nM T92057 D00NYJ 42642648 IC50 = 4 nM T92057 D02TUL 118115473 IC50 = 25200 nM T92057 D02UFQ 11620908 IC50 = 260 nM T92057 D03LWG 53235510 IC50 > 10000 nM T92057 D07EHV 44814409 IC50 > 10000 nM T92057 D07HPJ 11476171 IC50 = 1700 nM T92057 D0E3TC 44259 IC50 = 282 nM T92057 D0G5XV 135565884 IC50 = 1.58 nM T92057 D0QX8X 71479709 IC50 = 37.9 nM T92057 D0U4FF 10437018 IC50 = 190 nM T92057 D0YB3W 156414 IC50 = 10 nM T92057 D02YAQ 6603857 IC50 = 20 nM T92057 D0T3ME 156422 IC50 > 30000 nM T92057 CRFU83 156413 IC50 = 27 nM T92057 CPXK25 5793057 IC50 = 7740 nM T92057 CB7WK3 5938113 IC50 = 23900 nM T92057 C41QWA 9857146 IC50 > 10000 nM T92057 CW8V0K 9864418 IC50 > 25000 nM T92057 C01WSX 9907221 IC50 = 1.7 nM T92057 C37GXK 9983303 IC50 > 25000 nM T92057 C2C1BP 10089048 IC50 > 25000 nM T92057 CRX6F0 10479082 IC50 > 25000 nM T92057 CU27LB 11246488 IC50 = 49 nM T92057 CBOP58 11293798 Ki > 10000 nM T92057 C26BZX 11362471 Ki > 10000 nM T92057 CWXB93 11397177 Ki > 10000 nM T92057 C94QJA 11420204 IC50 = 66 nM T92057 C6-AUG 11496207 IC50 = 538 nM T92057 C08APU 11503073 IC50 = 229 nM T92057 CU13WV 11518389 IC50 = 1.2 nM T92057 CF0YW7 11518637 IC50 = 624 nM T92057 CV3NK7 11524106 IC50 = 7.1 nM T92057 CT75DZ 11532242 IC50 = 16 nM T92057 C5VO2C 11539461 IC50 = 6.2 nM T92057 CX6KD1 11553647 IC50 = 310 nM T92057 CKUR82 11568720 IC50 = 1 nM T92057 CN31OR 11590557 IC50 = 4.3 nM T92057 CR06MA 11595844 IC50 = 7.3 nM T92057 CR1FG0 11604864 IC50 = 1.8 nM T92057 C9T3VC 11613187 IC50 = 0.8 nM T92057 CG0K4A 11632391 IC50 = 2.4 nM T92057 CB4YR6 11634425 IC50 = 73 nM T92057 CA8X1L 11655791 IC50 = 59 nM T92057 C5J8NA 11703562 IC50 > 100 nM T92057 CXOF82 11711590 IC50 = 644 nM T92057 C4YWU2 11713043 IC50 = 1 nM T92057 C8WQ9F 11719423 IC50 = 11 nM T92057 CQF23E 11952856 IC50 = 11 nM T92057 CFPW41 16007116 Ki > 3800 nM T92057 CM2HS9 18176200 IC50 = 13 nM T92057 CA3I4T 24753787 IC50 > 50000 nM T92057 C61KPI 24856363 IC50 > 25000 nM T92057 C43HWQ 24883287 IC50 < 100 nM T92057 C8DA5Q 24883334 IC50 < 100 nM T92057 CG3XC9 25124150 IC50 = 74 nM T92057 CO2IR5 25124816 IC50 > 25000 nM T92057 CEL61X 44229839 IC50 = 79 nM T92057 CWFB42 44571820 IC50 = 140 nM T92057 C7Q1VU 44580077 IC50 > 25000 nM T92057 CL90SE 44580358 IC50 > 25000 nM T92057 CK1VE7 44580420 IC50 > 25000 nM T92057 CH2R7X 44580449 IC50 > 25000 nM T92057 C1VH0C 44580532 IC50 > 25000 nM T92057 CXC52J 44580649 IC50 > 25000 nM T92057 CE32BQ 44580689 IC50 = 300 nM T92057 C8Z5AX 44580778 IC50 > 25000 nM T92057 CY3HW5 46224684 IC50 > 10000 nM T92057 CLS29B 46872626 IC50 > 10000 nM T92057 C2O8RZ 46886323 IC50 = 18 nM T92057 C9PAT7 46927672 IC50 = 10 nM T92057 CEQN27 52936621 Ki > 1000 nM T92057 CQ87LD 52946569 IC50 = 50 nM T92057 CNPM14 53341082 IC50 = 4 nM T92057 CBK9Q6 53357848 IC50 > 10000 nM T92057 C8NA4L 53384644 IC50 > 30000 nM T92057 C1XS2J 54760383 IC50 = 30 nM T92057 CE1A9V 57394653 IC50 = 43.7 nM T92057 C10AMI 66553589 IC50 > 10000 nM T92057 CV63UL 67240318 IC50 > 10000 nM T92057 C8I7GC 68293638 IC50 > 10000 nM T92057 C7VJ6A 70647728 IC50 = 50 nM T92057 CQ5W6D 70693519 IC50 = 74 nM T92057 COU73Y 71226944 IC50 = 71 nM T92057 C40JOZ 71235465 IC50 = 169 nM T92057 CEBO91 71452977 IC50 = 160 nM T92057 CKT60L 71455860 Ki > 3700 nM T92057 C9DIK2 71512060 IC50 = 23 nM T92057 CRX81Q 71575642 IC50 > 10000 nM T92057 C1BCX0 71579696 IC50 > 1000 nM T92057 CZ31PU 71583657 IC50 = 240 nM T92057 CIU90H 72202607 IC50 = 3 nM T92057 C60TUV 72737208 IC50 = 12 nM T92057 CJ3WA6 72737404 IC50 = 8 nM T92057 CVNW01 73386831 IC50 > 1000 nM T92057 CDNQ20 73388819 IC50 = 11.3 nM T92057 CN39OQ 78341183 IC50 = 44 nM T92057 CCJ43A 86302281 IC50 = 4 nM T92057 CB5NJ4 86302541 IC50 > 10000 nM T92057 CPG3A5 86302574 IC50 > 30000 nM T92057 CX29IY 90655145 IC50 = 37 nM T92057 C37DUM 121293882 IC50 = 240 nM T92057 CXQR89 121294143 IC50 = 10 nM T92057 C4X7SD 122192466 IC50 > 10000 nM T92057 CKS28E 127034802 IC50 = 213 nM T92057 CKX40V 127037812 IC50 > 10000 nM T92057 C70RUP 127038480 IC50 > 10000 nM T92057 C3WCN8 127041777 IC50 > 10000 nM T92057 CP15ZX 127043295 IC50 = 801 nM T92057 CV0F3N 127045112 IC50 = 1100 nM T92057 CTPY32 127045266 IC50 = 930 nM T92057 CWI8Q2 127045267 IC50 = 782 nM T92057 CV5I8S 127045270 IC50 = 1603 nM T92057 CIU72D 127264586 IC50 = 3.2 nM T92057 CUO0C5 132156633 IC50 > 10000 nM T92057 CV89JM 132231876 IC50 = 150 nM T92057 CERS64 132937256 IC50 > 30000 nM T92057 CM5T6K 134130825 IC50 = 2 nM T92057 CC1EB5 134131929 IC50 = 6 nM T92057 CMZG34 134133313 IC50 = 2 nM T92057 CX2WN6 134134364 IC50 = 10 nM T92057 CSZX25 134135323 IC50 = 5 nM T92057 C1GVQ7 134136098 IC50 = 82 nM T92057 C3G7TQ 134136245 IC50 = 11 nM T92057 CJ7C1N 134137974 IC50 = 7 nM T92057 CY3U6V 134138310 IC50 = 460 nM T92057 C4QSZ5 134138566 IC50 = 13 nM T92057 CZU97C 134138682 IC50 = 3 nM T92057 C6RGN8 134138812 IC50 = 27 nM T92057 C58FUC 134139047 IC50 = 376 nM T92057 C6U5WE 134139490 IC50 = 15 nM T92057 CA7PD8 134139534 IC50 = 94 nM T92057 C3OBC6 134139548 IC50 = 94 nM T92057 CW69GT 134139694 IC50 = 4 nM T92057 CQE08L 134139702 IC50 = 302 nM T92057 C8JR1X 134140108 IC50 = 4 nM T92057 CY8UF9 134140285 IC50 = 213 nM T92057 C6UJG4 134140680 IC50 = 108 nM T92057 CI2L7Z 134140949 IC50 = 487 nM T92057 CY9M7L 134143068 IC50 = 653 nM T92057 CSTC29 134143257 IC50 = 40 nM T92057 C4F6VU 134143525 IC50 = 5 nM T92057 C38JMR 134145160 IC50 = 285 nM T92057 CO7LU3 134145579 IC50 = 64 nM T92057 C1OYR9 134145751 IC50 = 48 nM T92057 CKZ2I0 134145988 IC50 = 583 nM T92057 CRZ0E5 134146010 IC50 = 4 nM T92057 CTMJ14 134146542 IC50 = 97 nM T92057 CN35SO 134146628 IC50 > 1000 nM T92057 CHJ13S 134146699 IC50 = 4 nM T92057 C0KNV3 134146887 IC50 = 4 nM T92057 C4U8KT 134147234 IC50 = 6 nM T92057 CJ1FQ6 134147869 IC50 = 3 nM T92057 CXS38A 134147887 IC50 = 88 nM T92057 CPGL96 134148137 IC50 = 18 nM T92057 CGVC01 134148454 IC50 = 328 nM T92057 C5R2PK 134148588 IC50 = 29 nM T92057 C0AWH3 134148660 IC50 = 10 nM T92057 C6Z2JL 134149963 IC50 = 22 nM T92057 CE69LC 134150331 IC50 = 4 nM T92057 CJ56EZ 134150417 IC50 = 28 nM T92057 CRC81V 134150452 IC50 = 428 nM T92057 CQK40B 134150618 IC50 = 4 nM T92057 C7CT2Y 134151327 IC50 = 95 nM T92057 CI4A1T 134152401 IC50 = 41 nM T92057 C0N6JF 134152887 IC50 = 3 nM T92057 C9ORY0 134152991 IC50 = 38 nM T92057 CW6A7E 134153017 IC50 = 78 nM T92057 CLBK62 134153313 IC50 = 408 nM T92057 C6JFN5 134153988 IC50 = 4 nM T92057 C5YX7T 134154596 IC50 = 3 nM T92057 C07RWN 134154721 IC50 = 18 nM T92057 CV5M1T 134154754 IC50 = 1 nM T92057 CI0S4B 134155078 IC50 = 636 nM T92057 CMH0X4 134155167 IC50 = 514 nM T92057 C9DRQ6 134155700 IC50 = 4 nM T92057 C6HN5J 134155932 IC50 = 43 nM T92057 CQD93J 134156816 IC50 = 3 nM T92057 C3HCT6 134156845 IC50 = 3 nM T92057 CF85NI 134157315 IC50 = 676 nM T92057 CG36DX 134157614 IC50 = 63 nM T92057 CYL5V1 134694986 IC50 > 30000 nM T92057 C3Z4AT 137321159 IC50 > 10000 nM T92057 C25ERN 137631967 IC50 = 5 nM T92057 CZOD53 137633880 IC50 = 230 nM T92057 C7BJY5 137636807 IC50 = 76 nM T92057 C06JRX 137637094 IC50 = 6.2 nM T92057 C7TG3J 137641313 IC50 > 19952.62 nM T92057 CO89DX 137649100 IC50 = 59 nM T92057 C1DK0P 137651391 IC50 = 2.4 nM T92057 CINE03 137652514 IC50 = 514 nM T92057 C28QUP 137652864 IC50 = 1004 nM T92057 CV5H3Z 137657932 IC50 = 5.3 nM T92057 CSRI06 138547901 IC50 > 1000 nM T92057 CUXO19 138617501 IC50 > 1000 nM T92057 CO9P7G 145351804 IC50 > 1000 nM T92057 C29XUO 145945978 IC50 > 1000 nM T92057 C3LW9D 145952066 IC50 = 6400 nM T92057 C6G4NF 145955071 IC50 = 4410 nM T92057 CLK9N3 145959197 IC50 = 6430 nM T92057 CHT30M 145959430 IC50 = 8050 nM T92057 CMC76F 145959984 IC50 = 5060 nM T92057 C4OD9Q 145967187 IC50 = 0.6 nM T92057 CE31VG 145979714 IC50 > 10000 nM T92057 C9BX4U 145988956 IC50 = 3540 nM T92057 C2MD1Q 155513187 IC50 > 10000 nM T92057 C86HPW 155518524 IC50 = 7900 nM T92057 C3NA2I 155519537 IC50 = 385 nM T92057 C78MZC 155536330 IC50 = 3 nM T92057 CE46SL 155540854 IC50 = 4680 nM T92057 C5O4JM 155540856 IC50 = 1500 nM T92057 CGVU70 155554426 IC50 = 29020 nM T92057 D00ERW 44444843 Ki > 3750 nM T92057 D00TZD 2776 IC50 = 12 nM T92057 D01RHR 71519693 IC50 = 5.5 nM T92057 D01VFR 4708 IC50 = 12 nM T92057 D03BJB 9549299 IC50 = 7640 nM T92057 D05FFT 11566580 IC50 = 0.5 nM T92057 D06BJG 71556703 IC50 = 3.3 nM T92057 D0D6MH 11617559 IC50 > 24000 nM T92057 D0Q0YV 24944925 IC50 > 19952.62 nM T16263 CX5V7B 50898694 IC50 = 32 nM T16263 C9M0KE 52941821 IC50 = 23 nM T16263 CJ3D7Y 52941822 IC50 = 38 nM T16263 CI3C8V 52942058 IC50 = 27 nM T16263 CLO38X 52942071 IC50 = 25 nM T16263 C2G1RT 52942078 IC50 = 102 nM T16263 C5VDS7 52942148 IC50 = 27 nM T16263 C9G8VW 52943283 IC50 = 47 nM T16263 C86MFB 52944231 IC50 = 215 nM T16263 CQ38KM 52944537 IC50 = 35 nM T16263 C64CAT 52944644 IC50 = 40 nM T16263 C4KLV6 52945332 IC50 = 17 nM T16263 CLAH27 52946506 IC50 = 27 nM T16263 C07PSZ 52946910 IC50 = 22 nM T16263 CG8S9O 52946946 IC50 = 32 nM T16263 CA7Z6L 52946953 IC50 = 72 nM T16263 C1C5BV 52946954 IC50 = 31 nM T16263 CY1BP4 52947004 IC50 = 52 nM T16263 C1X9RI 52947038 IC50 = 39 nM T16263 C0F1WE 52947044 IC50 = 35 nM T16263 CKI5X6 52947100 IC50 > 500 nM T16263 C1ZK2O 52947741 IC50 > 500 nM T16263 CJT61Q 52947748 IC50 = 23 nM T16263 C2V4EQ 52948136 IC50 = 25 nM T16263 C2S7HO 52948142 IC50 = 25 nM T16263 CZK6D2 52948162 IC50 = 68 nM T16263 C64DXZ 52948248 IC50 > 500 nM T16263 CKS2T4 52949127 IC50 = 48 nM T16263 CI5EM7 52949128 IC50 = 104 nM T16263 CU25FT 52949601 IC50 = 207 nM T92777 D04ZTY 444020 IC50 = 1300 nM T92777 D0D0ZD 441314 Ki = 1000 nM T92777 D0HR8Z 51634 IC50 = 2100 nM T92777 D0MU9L 176077 IC50 = 1500 nM T92777 D07TSW 6451151 Ki = 1000 nM T92777 D0L4FS 5280961 IC50 = 2610 nM T92777 D0RE9C 501391 IC50 = 10000 nM T92777 D0S5LT 29435 IC50 = 360 nM T92777 CR8UX7 2859 IC50 < 100000 nM T92777 CG0YT4 92381 IC50 = 120 nM T92777 CO8GW2 193758 IC50 = 100000 nM T92777 CDR69S 195553 Ki = 6200 nM T92777 CBJ30L 444254 IC50 = 906000 nM T92777 C9PU8M 446685 IC50 = 110000 nM T92777 CVMQ20 451990 IC50 < 50000 nM T92777 C71DGH 451992 IC50 = 500000 nM T92777 C50GBF 464727 IC50 < 50000 nM T92777 C6Y9MV 464728 IC50 < 50000 nM T92777 C6NIV0 6475028 IC50 = 8400 nM T92777 CVT72N 6475029 Ki = 450 nM T92777 C8P1VD 6475031 IC50 = 4200 nM T92777 C7UIV5 6477160 IC50 = 60 nM T92777 CQ1Z0B 9883791 Ki = 1000 nM T92777 C0VWI8 10039088 Ki = 2.3 nM T92777 CAWL97 10888248 IC50 > 1000000 nM T92777 C06FUY 11105683 IC50 > 1000000 nM T92777 CC4N0X 11258014 IC50 > 500000 nM T92777 C9D5WG 11547355 IC50 > 100 ug.mL-1 T92777 CGE87W 11630203 IC50 = 550 nM T92777 CFWZ59 11640963 IC50 = 16000 nM T92777 C3V0EP 11748894 IC50 = 9000 nM T92777 C1JBA9 11816841 IC50 > 1000000 nM T92777 CR3J0F 13076018 IC50 < 100000 nM T92777 C7UOT0 15218073 Ki = 2500 nM T92777 CA63TV 15218074 Ki = 2600 nM T92777 C8K0JT 15221166 Ki = 50 nM T92777 CJ14DK 15221167 Ki = 120 nM T92777 CZD64F 15389573 Ki = 900 nM T92777 C1WA3T 15389574 Ki = 10000 nM T92777 C1GO6Q 15389575 Ki = 28 nM T92777 C3IJ4O 16121613 IC50 = 58000 nM T92777 C3V0ON 16121614 IC50 = 82000 nM T92777 COHX16 16196970 IC50 > 100 ug.mL-1 T92777 C0NW5L 21021619 IC50 = 17000 nM T92777 CZ21NH 23622616 IC50 > 1000000 nM T92777 CCV9J1 25010555 Ki = 100 nM T92777 CET6K7 25010557 Ki = 130 nM T92777 C4GUL0 44346057 Ki = 87 nM T92777 CTLZ02 44346152 Ki = 4 nM T92777 CG61EN 44346204 Ki = 10 nM T92777 CDV7C9 44346217 Ki = 70 nM T92777 C02QTR 44384023 IC50 < 100000 nM T92777 C5TPW9 44384057 IC50 = 50000 nM T92777 C2QGH7 44411113 IC50 = 100000 nM T92777 CFV89K 44411114 IC50 = 120000 nM T92777 COZ73Y 44411115 IC50 = 101000 nM T92777 CCNH25 44411124 IC50 = 110000 nM T92777 CYU46L 44411131 IC50 = 101000 nM T92777 CI2UA7 44411422 IC50 = 58000 nM T92777 CP43TZ 44437482 IC50 = 84000 nM T92777 CY9XI2 44437483 IC50 = 70000 nM T92777 C7SI6M 44437486 IC50 = 100000 nM T92777 CO2A3P 44437487 IC50 = 28000 nM T92777 CSZW17 44437488 IC50 = 16000 nM T92777 CCY45T 44437489 IC50 = 6000 nM T92777 CY1I4N 44437490 IC50 = 14000 nM T92777 CNH46K 44437491 IC50 = 25000 nM T92777 CTQ30E 44437492 IC50 = 36000 nM T92777 C1S8XD 44437493 IC50 = 11000 nM T92777 CYN5E2 44514060 Ki = 80 nM T92777 C6B2SM 44514354 Ki = 60 nM T92777 C9XN1W 44559227 IC50 > 100 ug.mL-1 T92777 CQ3SX9 44820249 IC50 = 15000 nM T92777 CNL06X 44820252 IC50 > 1000000 nM T92777 CKE7T2 45139324 Ki = 20 nM T92777 CLI3J7 46187831 Ki = 43 nM T92777 CQ28NZ 46187833 Ki = 15 nM T92777 C0UPQ4 46861742 Ki = 200 nM T92777 C9QVG2 46945258 Ki = 500 nM T92777 CB01CN 52944669 Ki = 1400 nM T92777 C3UTM6 54580834 IC50 = 960 nM T92777 C1I9YL 54584900 IC50 = 100000 nM T92777 C4ROH9 54586701 IC50 = 1100 nM T92777 CKL6U4 54587740 IC50 = 2000 nM T92777 CPEZ95 60201905 IC50 = 150 nM T92777 C6MPS3 70682078 IC50 = 3200 nM T92777 CLD7G4 70684192 IC50 = 7200 nM T92777 C3CT8H 70688441 IC50 = 650 nM T92777 C7DM2F 70688442 IC50 = 68 nM T92777 CK41SJ 70688446 IC50 = 1500 nM T92777 CT3DW5 70690487 IC50 = 100000 nM T92777 CV0LZ5 70690489 IC50 = 4.9 nM T92777 C7WK3N 70692637 IC50 = 100 nM T92777 C9TFL7 70692640 IC50 = 80000 nM T92777 C1GF6S 70694681 IC50 = 28 nM T92777 CK0HZ7 70694688 IC50 = 70 nM T92777 CPI7U6 70696726 IC50 = 72 nM T92777 CDC84M 73347264 IC50 = 34000 nM T92777 C5TU1M 73350356 IC50 = 5.8 nM T92777 CM81IL 73356409 IC50 = 13 nM T92777 C6CZ0Y 73356410 IC50 = 5000 nM T92777 CJ0C5O 101872894 IC50 = 6.1 nM T92777 C2NXA4 101882899 IC50 = 9000 nM T92777 C05DUA 101882900 IC50 > 100000 nM T92777 CH5U7F 118411068 IC50 = 7000 nM T92777 C8X6RN 118411069 IC50 > 100000 nM T92777 C16QGB 118411070 IC50 > 100000 nM T92777 CD76NI 118411071 IC50 = 8000 nM T92777 C9LGB3 118411072 IC50 = 2500 nM T92777 CAR82K 118411073 IC50 = 2000 nM T92777 CGXZ37 118411074 IC50 = 3000 nM T92777 C8G3LO 118411076 IC50 = 1500 nM T92777 CB72ZY 118411077 IC50 > 100000 nM T92777 C2CF0W 118411108 IC50 > 100000 nM T92777 CH7BA2 118411149 IC50 > 100000 nM T92777 CUYO63 118411153 IC50 > 100000 nM T92777 CK4EY8 118718367 IC50 = 15 nM T92777 C0CB8Y 118718368 IC50 = 240 nM T92777 C1Q5LO 118718369 IC50 = 410 nM T92777 C7UZH5 118718370 IC50 = 230 nM T92777 C4UFL8 118718371 IC50 = 5900 nM T92777 C1FY0J 118718372 IC50 = 100 nM T92777 CQ97ZM 118718373 IC50 = 520 nM T92777 CWX6I0 118718374 IC50 = 1600 nM T92777 CVM9B6 118718375 IC50 = 200 nM T92777 CR74KA 118718376 IC50 = 43 nM T92777 CN60OK 118718377 IC50 = 270 nM T92777 C5I7KQ 118718379 IC50 = 330 nM T92777 CC8N6I 118719919 IC50 = 1500 nM T92777 C1WON3 118720302 IC50 = 2500 nM T92777 C0ZOT7 118720303 IC50 = 4000 nM T92777 C81YUI 118720304 IC50 > 100000 nM T92777 CXI04D 118720305 IC50 > 100000 nM T92777 CG7JV9 118720306 IC50 > 100000 nM T92777 CR4S5Y 118720307 IC50 > 100000 nM T92777 CG9Q8E 118720308 IC50 > 100000 nM T92777 C7WD2O 118730249 IC50 = 10230 nM T92777 C93PLI 118730252 IC50 = 8480 nM T92777 CWO19P 118730256 IC50 = 12750 nM T92777 C1HX3G 118730261 IC50 = 26380 nM T92777 C39VNJ 118730263 IC50 = 7120 nM T92777 CTV27Y 118730264 IC50 = 16170 nM T92777 C9NPI5 118730265 IC50 = 8050 nM T92777 C07QMC 118730266 IC50 = 28020 nM T92777 CCDH86 118730267 IC50 = 18330 nM T92777 C0L5SN 118730270 IC50 = 5310 nM T92777 CHJ12O 118730271 IC50 = 11090 nM T92777 C8UC7H 118730272 IC50 = 9210 nM T92777 CAR5H4 118730275 IC50 = 44800 nM T92777 C4AC0G 118730277 IC50 = 11120 nM T92777 CJA0L7 127048314 IC50 = 470 nM T92777 C9DEI5 127051169 IC50 = 690 nM T92777 C2R3UJ 127052422 IC50 = 1500 nM T92777 CSO12K 127052423 IC50 = 640 nM T92777 CXV8U5 136180344 IC50 = 8370 nM T92777 C4V1RS 136961465 IC50 = 6500 nM T92777 C90LJD 136961466 IC50 = 11290 nM T92777 CCUO70 136961467 IC50 = 11220 nM T92777 C53NIY 136961468 IC50 = 6970 nM T92777 CMR4O0 136961469 IC50 = 5550 nM T92777 C35CJD 136961470 IC50 = 15090 nM T92777 C08YHA 136961471 IC50 = 5580 nM T92777 C1JZ2Y 136961472 IC50 = 8070 nM T92777 COLK97 136961473 IC50 = 53340 nM T92777 CVA54E 136961474 IC50 = 11850 nM T92777 CX0K8W 145948806 IC50 = 15200 nM T92777 C0NO6V 44514062 Ki = 90000 nM T92777 CHMN60 52941050 Ki = 2300 nM T92777 D03TYC 159496 IC50 = 40 nM T92777 D05GYF 11710941 Ki = 170 nM T92777 D08TQA 174312 IC50 = 2200 nM T92777 D0F9YZ 42632210 Ki = 190 nM T92777 D0GS0O 451991 IC50 = 55000 nM T92777 D0N9IX 9822159 IC50 = 3000 nM T92777 D0Q1KL 44320078 IC50 = 700 nM T92777 D0R5HV 124702 IC50 < 50000 nM T92777 D0W8GU 52942310 Ki = 30 nM T88547 D00HPK 47641 Ki = 880 nM T88547 D01AZG 5073 Ki = 4300 nM T88547 D01JUF 5775 IC50 = 549.54 nM T88547 D01XBA 5035 Ki = 38 nM T88547 D01ZSO 4235 Ki > 100 nM T88547 D02KRS 2130 Ki = 20.25 nM T88547 D03HFG 5324346 Ki = 36 nM T88547 D03QGM 5355 IC50 > 10000 nM T88547 D03SKD 5284603 Ki > 10000 nM T88547 D04XPW 446220 Ki = 8830 nM T88547 D06XMU 6013 Ki = 1200 nM T88547 D07BSQ 5994 Ki = 260 nM T88547 D07KSG 2733526 Ki = 35 nM T88547 D08VRO 3822 IC50 = 1 nM T88547 D09OBB 5360696 Ki = 348 nM T88547 D09VBC 2562 Ki = 19.5 nM T88547 D0CT9Y 1548953 Ki = 8 nM T88547 D0D1AL 3559 Ki = 0.2 nM T88547 D0D7TB 9417 Ki = 0.2 nM T88547 D0E1WI 3345 IC50 = 354 nM T88547 D0G8NN 119570 Ki = 4446 nM T88547 D0H6QU 6005 IC50 > 10000 nM T88547 D0H8QL 4020 IC50 = 234.42 nM T88547 D0I0DL 3689 IC50 = 3.9 nM T88547 D0K0TC 68617 Ki = 57 nM T88547 D0L5WM 2157 Ki = 1 nM T88547 D0M8VE 71360 IC50 = 64 nM T88547 D0NS6H 3152 Ki = 14.6 nM T88547 D0P6UB 10836 Ki = 8320 nM T88547 D0R4OM 5566 Ki = 15 nM T88547 D0T8GD 89594 IC50 > 10000 nM T88547 D0TR5X 3386 IC50 = 851.14 nM T88547 D0U2OO 2477 IC50 = 36.31 nM T88547 D0WE3O 5288826 Ki > 10000 nM T88547 D0X3FX 5284596 IC50 > 100000 nM T88547 D0Z1RV 135398737 Ki = 8500 nM T88547 D0Z6ST 2467 Ki = 1290 nM T88547 D00POS 9931976 Ki = 451 nM T88547 D00WLO 3455 IC50 = 43 nM T88547 D0A7KI 3037308 Ki = 490 nM T88547 D0I8FV 5567 Ki = 0.83 nM T88547 D0N1HW 5311200 Ki = 130 nM T88547 D0P1YE 9852175 Ki = 940 nM T88547 D0R8GR 9892540 IC50 = 47 nM T88547 D00KVE 9907323 Ki = 3.162 nM T88547 D0K6NS 6536 Ki = 8 nM T88547 D0H2SE 118607347 Ki = 23 nM T88547 D0N6JH 24968535 Ki = 1437 nM T88547 D0W3TS 41306362 Ki = 3.2 nM T88547 D00EZE 3047810 Ki = 19 nM T88547 D00ZGA 9917021 Ki = 2980 nM T88547 D01KIU 126402 Ki = 46.5 nM T88547 D01PIL 54477 Ki = 55 nM T88547 D01YOC 108046 Ki = 71 nM T88547 D02KLW 180081 IC50 > 10000 nM T88547 D07KYU 9330 Ki > 1000 nM T88547 D07ODD 132891 Ki > 6270 nM T88547 D08AWI 11430856 Ki = 100 nM T88547 D09DRG 9952420 IC50 = 1.3 nM T88547 D0M9GE 53389 IC50 = 450 nM T88547 D0OC3J 5281881 IC50 = 2.239 nM T88547 D0XK2K 9829526 Ki = 17 nM T88547 D0Z4QV 121967 Ki = 10 nM T88547 C5H0QN 1235 Ki = 59.7 nM T88547 C5IOL8 4910 Ki = 17 nM T88547 CW56ZA 5290 Ki = 269 nM T88547 C1WK2E 5417 Ki = 2.5 nM T88547 CE41ZK 7594 IC50 = 397 nM T88547 CP0O8I 9513 Ki = 309 nM T88547 CZC17M 9669 Ki = 36.5 nM T88547 C5VS0H 10098 Ki > 100000 nM T88547 CVW5J9 10220 Ki = 106 nM T88547 CTC8N0 14657 IC50 > 100000 nM T88547 C5EO7I 22648 IC50 = 2200 nM T88547 CM4VK9 33142 Ki = 27.7 nM T88547 CNZD18 36381 Ki = 30.1 nM T88547 C8Y6DE 37461 IC50 = 52.48 nM T88547 CO6M2K 41011 Ki = 3.1 nM T88547 CTF7Z4 50266 Ki = 230 nM T88547 CY2F8T 55445 IC50 = 76 nM T88547 C0RV1Y 60840 IC50 = 2540 nM T88547 C8CZ1E 64600 IC50 = 5 nM T88547 C0LQ7N 65638 Ki = 1 nM T88547 CLY10I 65659 Ki > 100 nM T88547 CDQX62 66270 Ki > 800 nM T88547 C0SKG4 66749 IC50 = 1250 nM T88547 C3WKC6 68835 IC50 = 27200 nM T88547 CZ6G7B 69873 Ki = 1980 nM T88547 CY79XW 72027 Ki = 4 nM T88547 C13JOV 75994 Ki = 10480 nM T88547 C34VIY 77042 IC50 > 5000 nM T88547 C0QAT3 88747 Ki > 10000 nM T88547 CB3U0P 90748 Ki = 0.67 nM T88547 CN26SL 93365 Ki = 0.01 nM T88547 C3JXH7 97478 Ki = 1150 nM T88547 CI8KD2 97627 Ki = 1480 nM T88547 CA3W0P 100826 IC50 > 100000 nM T88547 CY65GC 112416 IC50 > 10000 nM T88547 CW0G3U 119010 IC50 = 56 nM T88547 CM34NA 119265 Ki = 14.34 nM T88547 CT2H5A 121180 IC50 = 362 nM T88547 C21KTQ 121968 Ki = 10 nM T88547 CKR4N3 122065 Ki > 50 nM T88547 C1B4NI 125328 Ki = 2.4 nM T88547 CRJ7G1 126229 Ki = 0.9 nM T88547 C4VK3Y 126260 IC50 = 1.175 nM T88547 CYJ07C 126388 Ki = 0.34 nM T88547 C9BYH2 128032 Ki = 4.3 nM T88547 CE75MR 131253 Ki = 2 nM T88547 CNO1J3 131444 Ki = 17 nM T88547 CU0C6S 131698 Ki = 2.7 nM T88547 CUYI35 132954 IC50 = 3.47 nM T88547 C2KAL0 132995 Ki = 1.7 nM T88547 C85AXM 164487 IC50 = 26 nM T88547 C7QCS6 185717 IC50 = 50 nM T88547 C3SG4X 185834 Ki = 0.04 nM T88547 CFAP45 190868 Ki = 0.05 nM T88547 CNJ78I 192277 IC50 = 3020 nM T88547 CZDX91 192370 Ki = 168 nM T88547 C9Z3NL 192481 Ki = 10.4 nM T88547 CI9E2D 192611 IC50 = 0.29 nM T88547 CA3T7R 192638 IC50 = 228 nM T88547 CD19AW 192639 IC50 = 33 nM T88547 C5KHP9 200601 Ki = 5.81 nM T88547 CU2RH4 202478 Ki = 6 nM T88547 CDM25N 230867 IC50 > 10000 nM T88547 CF16XZ 242976 IC50 = 1370 nM T88547 C9EHT7 252230 IC50 = 15 nM T88547 C39OMI 269722 Ki = 5850 nM T88547 C0PUC2 344343 IC50 = 133 nM T88547 CZEG20 356862 IC50 = 2005 nM T88547 C30GUQ 381254 Ki = 1.64 nM T88547 C0DE9F 381255 Ki = 3.02 nM T88547 C5D4YG 398371 Ki = 720 nM T88547 C5JG2Z 398373 Ki = 2230 nM T88547 C13BVL 398418 Ki = 1100 nM T88547 CW0DY3 398578 Ki = 1.49 nM T88547 CXO6I9 398580 Ki = 1122 nM T88547 C7D0YB 398582 Ki = 77.5 nM T88547 C7QE8N 398586 Ki = 13.8 nM T88547 C01HIV 398588 Ki = 8 nM T88547 C3ZF6U 398839 Ki = 869 nM T88547 CM71EX 401804 Ki = 2220 nM T88547 C9AOD7 401806 Ki = 5460 nM T88547 C95KEG 401808 Ki = 3100 nM T88547 CNAU07 401810 Ki = 276 nM T88547 C3I7AM 401812 Ki = 291 nM T88547 CZLP87 401816 Ki = 579 nM T88547 C7EIT9 401818 Ki = 56 nM T88547 C29XHP 401820 Ki = 26 nM T88547 CH35LT 401822 Ki = 13 nM T88547 CCF24R 401826 Ki = 8.2 nM T88547 C27VBR 401827 Ki = 2.2 nM T88547 CM8JT4 401829 Ki = 1.3 nM T88547 C3AJZ6 401834 Ki = 3.9 nM T88547 CF1IA7 401839 Ki = 1.3 nM T88547 CTMQ39 401843 Ki = 148 nM T88547 CA93IJ 401844 Ki = 4.1 nM T88547 C43UDC 401846 Ki = 2.6 nM T88547 C6KN4X 401850 Ki = 4.1 nM T88547 CM57RI 401854 Ki = 4.8 nM T88547 C8JQ0S 401856 Ki = 2 nM T88547 CD9UV5 401860 Ki = 3.9 nM T88547 C1WEY2 401862 Ki = 1.4 nM T88547 CIX84S 407725 IC50 = 48 nM T88547 C7UEP4 409922 Ki = 7.6 nM T88547 C3HFE4 422923 Ki = 74 nM T88547 CCO6D8 428911 IC50 = 340 nM T88547 C4Y0ME 442108 Ki = 8554 nM T88547 C90GUY 473059 Ki = 72 nM T88547 C06MHS 473073 Ki = 47 nM T88547 CVZ3N0 547467 Ki = 2.3 nM T88547 CB8J6E 558800 Ki = 1.47 nM T88547 CKI0U2 558843 Ki = 4.22 nM T88547 C6AVL5 566741 Ki = 3.69 nM T88547 C4GF6U 573546 Ki = 2.67 nM T88547 CRMK45 573661 Ki = 3.56 nM T88547 CTW61R 574780 Ki = 6.3 nM T88547 CX5W2H 587944 Ki = 0.31 nM T88547 C5P9MF 594236 Ki = 0.39 nM T88547 C1Q3GW 604376 Ki = 0.52 nM T88547 C82CBK 620985 IC50 = 83 nM T88547 CJL68V 648525 IC50 = 1480 nM T88547 C35WDY 659840 Ki = 26 nM T88547 CQD2N8 728567 IC50 = 3500 nM T88547 C74ZXL 743379 Ki = 6.7 nM T88547 CU1R0C 762654 Ki = 11360 nM T88547 C80NWF 762919 Ki = 0.47 nM T88547 CQJW96 763622 Ki = 0.39 nM T88547 CRBO37 764022 Ki = 0.58 nM T88547 CUE5T3 764613 Ki = 1.4 nM T88547 CTF1D3 764825 Ki = 5.3 nM T88547 CM6Z0W 765219 Ki = 0.46 nM T88547 C8HU1D 782728 Ki = 706 nM T88547 C5S3MB 785789 Ki = 3.8 nM T88547 CUF0O4 796534 IC50 = 109 nM T88547 CS4XQ9 1081502 Ki > 100 nM T88547 CK04FA 1245023 Ki = 6.46 nM T88547 CK0JI9 1548955 Ki = 5 nM T88547 CUF6Z2 2225138 Ki = 26.9 nM T88547 CT7GF8 2427316 Ki = 0.2089 nM T88547 CHA7K3 2712605 Ki = 3.93 nM T88547 CLU95O 2729533 Ki = 30.8 nM T88547 C8VTI5 2817997 Ki = 3.9 nM T88547 CF96BK 2845469 Ki = 10.5 nM T88547 CZ7C0Q 2845594 Ki = 7.5 nM T88547 C9FHM1 3035672 Ki = 0.8 nM T88547 CM3GY5 3036027 Ki = 1.3 nM T88547 C2TAD3 3036289 Ki = 696 nM T88547 C4TB0I 3036864 IC50 = 389.05 nM T88547 CZPH80 3037711 Ki = 82.9 nM T88547 CLB7W5 3037886 Ki = 2100 nM T88547 CE4KC8 3038603 Ki = 800 nM T88547 C54FEG 3039881 Ki = 550 nM T88547 C7MQC0 3041078 Ki = 482 nM T88547 C6RJ5X 3043720 Ki = 22 nM T88547 C6Z4QI 3050372 Ki = 77.1 nM T88547 CI5W4L 3064081 IC50 > 10000 nM T88547 C5NA6S 3069135 Ki = 41.5 nM T88547 CJ7K3Y 3081049 Ki = 3720 nM T88547 CNL68D 3083456 IC50 = 4 nM T88547 C2SE0V 3083457 IC50 = 0.5 nM T88547 CS5F1I 3083481 Ki = 4.4 nM T88547 C6AX8Y 3126148 Ki > 100 nM T88547 C0WFU5 3296345 Ki = 66.4 nM T88547 CJ4Y7Q 3299322 Ki = 2.9 nM T88547 C6G4UP 3315413 IC50 = 140 nM T88547 CJ6D8N 3342390 Ki < 1000 nM T88547 C7V3QI 3562491 Ki = 22.66 nM T88547 CE49MQ 3869448 Ki = 1.46 nM T88547 CGUE70 4033090 Ki = 6.65 nM T88547 CW9SC1 4058484 IC50 > 10000 nM T88547 CWX41S 4598397 Ki = 12 nM T88547 CRM98I 4687238 IC50 = 0.7244 nM T88547 CO84FU 4827344 Ki = 9.66 nM T88547 C47FSG 4879851 Ki = 10.1 nM T88547 CO30PB 4992580 Ki = 19.2 nM T88547 CZF7B5 5026275 Ki = 0.17 nM T88547 C2M4DQ 5221975 Ki = 3.9 nM T88547 C4J7FP 5236783 Ki = 4.89 nM T88547 CK8D2C 5370189 Ki = 0.86 nM T88547 CR4G2N 5461916 Ki = 0.67 nM T88547 C95ADL 5468874 Ki = 7436 nM T88547 CVCA38 5468876 Ki = 27.3 nM T88547 C2DNO0 5471948 Ki = 2.4 nM T88547 C97VGU 5474589 Ki = 3 nM T88547 C0J2GT 5478726 Ki = 1.3 nM T88547 C6ZL2O 5974189 IC50 = 51 nM T88547 CFGZ19 6273133 Ki = 3.2 nM T88547 CB3M8S 6331636 Ki = 455 nM T88547 C9J6HG 6430604 Ki = 275 nM T88547 CFO08L 6437849 Ki = 680 nM T88547 C2UV7A 6439331 Ki = 3 nM T88547 CIPW27 6465840 Ki = 30.1 nM T88547 CGM63Y 6540428 IC50 = 912.01 nM T88547 CED0X6 6604724 Ki = 594 nM T88547 C5WH0F 6604868 IC50 = 28 nM T88547 C6R4WZ 6712729 Ki = 11.2 nM T88547 CCU3H5 6712751 IC50 = 278 nM T88547 C9G5RB 6712752 IC50 = 128 nM T88547 C1M9QS 6713949 Ki = 81 nM T88547 C0S1MT 6918656 Ki = 4.3 nM T88547 C1ORF3 6995232 Ki = 1258.93 nM T88547 C4Z0DT 9049339 Ki = 2.1 nM T88547 CCN7X5 9208936 Ki = 3.97 nM T88547 C9UB2N 9795762 Ki = 10 nM T88547 C4V0PN 9796317 Ki = 5.4 nM T88547 C24EXG 9796923 Ki = 0.51 nM T88547 CK3DI8 9797419 Ki = 6.59 nM T88547 CNXS47 9797436 Ki = 1.39 nM T88547 CDT7Q4 9797984 IC50 = 10700 nM T88547 CD8H3W 9799239 Ki = 0.5 nM T88547 CPB9S2 9800653 IC50 = 7551 nM T88547 CXI46Z 9802946 Ki = 13.82 nM T88547 C32AXD 9803895 Ki = 2.25 nM T88547 C7R0UJ 9804703 Ki = 3.21 nM T88547 CN2XR0 9817442 IC50 = 54 nM T88547 C0XJ8E 9817503 IC50 = 5.888 nM T88547 C2FVL8 9818804 IC50 = 16 nM T88547 CWJB39 9819510 Ki = 6.3 nM T88547 CJ96KD 9820591 Ki = 4.4 nM T88547 CH60LU 9823429 IC50 = 1.8 nM T88547 C82CXQ 9835629 IC50 = 1860 nM T88547 C73NUA 9835807 IC50 = 362 nM T88547 C5EDO7 9839491 Ki = 1 nM T88547 C9PC6E 9839973 IC50 = 2190 nM T88547 CHSR07 9840044 Ki = 56 nM T88547 C26QDV 9840310 Ki = 8.22 nM T88547 CXYJ93 9841596 Ki = 1 nM T88547 C89FSJ 9841846 Ki = 1.15 nM T88547 C3FK5G 9847317 Ki = 81 nM T88547 C6CXW8 9858146 IC50 = 1210 nM T88547 C17IQN 9861694 Ki = 4.3 nM T88547 CGC5E7 9862757 IC50 = 1000 nM T88547 CTF7N5 9863340 Ki = 2 nM T88547 C0BQA3 9864023 Ki = 14 nM T88547 CBW2I4 9864749 Ki = 0.67 nM T88547 C5XBP1 9868470 Ki = 4.2 nM T88547 C2V9FQ 9882367 Ki = 1.11 nM T88547 CAI67X 9882743 Ki = 654 nM T88547 CX8M6A 9883221 Ki = 2 nM T88547 C40DMV 9883360 Ki = 0.26 nM T88547 CX9P2S 9883361 Ki = 1.48 nM T88547 CI2R9W 9883362 Ki = 0.83 nM T88547 CL5V6S 9883820 Ki = 10.16 nM T88547 C3DB5H 9884781 Ki = 1.6 nM T88547 CTAC24 9885114 Ki = 232 nM T88547 CP1GD3 9887523 Ki = 1.21 nM T88547 C2S8KJ 9889112 Ki = 6.75 nM T88547 CA7F6X 9889113 Ki = 9.03 nM T88547 CHB63J 9889709 Ki = 4.8 nM T88547 CTY4K6 9890959 IC50 = 43 nM T88547 CL0Z7Q 9902485 IC50 = 6130 nM T88547 CNO38Q 9905222 Ki = 7 nM T88547 C4UP3E 9905985 Ki = 0.49 nM T88547 CH7K4W 9906138 Ki = 5.51 nM T88547 CAEG95 9906139 Ki = 3.15 nM T88547 CYWQ50 9906447 Ki > 10000 nM T88547 C9XIG6 9919363 IC50 = 13 nM T88547 C7PC1V 9921810 IC50 = 82 nM T88547 C0UH2P 9923341 IC50 = 4800 nM T88547 CY3FW6 9924349 Ki = 3.3 nM T88547 CV28TC 9925741 Ki = 0.25 nM T88547 C85CAL 9926814 Ki = 0.98 nM T88547 CAY53L 9927364 Ki = 3.56 nM T88547 CS29LN 9927617 Ki = 1300 nM T88547 CBSW20 9930604 Ki = 288.4 nM T88547 C1UA3Y 9936242 Ki = 1.78 nM T88547 CSH40U 9936494 IC50 = 183 nM T88547 CN59VH 9943903 IC50 = 2.754 nM T88547 C78DMI 9951886 Ki = 1.3 nM T88547 CZ0AT6 9954083 Ki = 1 nM T88547 CIT01A 9956313 IC50 > 100 nM T88547 CKMW59 9957260 Ki = 110 nM T88547 CNB8Q5 9966844 IC50 = 6260 nM T88547 CDR7Y4 9970628 IC50 = 2900 nM T88547 C9OM2Z 9973696 Ki = 1.75 nM T88547 CPY61E 9973880 Ki = 40.7 nM T88547 CUHA14 9974013 IC50 = 965 nM T88547 CFSR80 9975973 IC50 = 52 nM T88547 C5VNI2 9981159 Ki = 66.2 nM T88547 CIP7Q9 9992101 Ki = 0.07 nM T88547 CFE9H1 9994390 IC50 = 2700 nM T88547 CE3HF7 9995041 IC50 = 240 nM T88547 C4CYX9 9996818 IC50 = 2290 nM T88547 C5AO4D 9998085 Ki = 4 nM T88547 C6WY0U 9999116 Ki = 21.6 nM T88547 C9T0UJ 9999184 IC50 = 320 nM T88547 CXU2V1 10001045 Ki = 128 nM T88547 C6QPD3 10001759 Ki = 76.9 nM T88547 CIZ3D8 10001888 Ki = 110 nM T88547 CX36LV 10002293 Ki = 0.65 nM T88547 CQ5NZ7 10016031 IC50 = 351 nM T88547 C97KHW 10017418 Ki = 2.7 nM T88547 CQH60R 10017724 Ki = 16.05 nM T88547 CG0IW7 10017936 Ki = 0.6 nM T88547 C1XK9Y 10019102 Ki = 1.29 nM T88547 C9LC6Z 10020651 IC50 = 140 nM T88547 C94EDH 10021099 Ki = 2 nM T88547 CQ9M7E 10021279 Ki = 2.5 nM T88547 C7HU5C 10021562 IC50 = 54.4 nM T88547 CS83XQ 10022628 Ki = 46 nM T88547 CFB0D2 10023021 Ki = 3.11 nM T88547 C3RH0Z 10023073 Ki = 0.87 nM T88547 CU93MX 10023529 Ki = 0.46 nM T88547 CL5IW1 10024634 Ki = 1.34 nM T88547 CB5T9V 10025360 IC50 = 1034 nM T88547 CSI9J6 10025403 Ki = 6.9 nM T88547 CI92JG 10025852 Ki = 16.53 nM T88547 CF6O3E 10027435 Ki = 2 nM T88547 CXZ3Q6 10037913 IC50 = 6280 nM T88547 C3S0HG 10037914 IC50 = 247 nM T88547 CFAO01 10038412 IC50 = 7180 nM T88547 C3Z4OD 10040286 Ki = 12 nM T88547 CZ2IY1 10041139 IC50 = 92 nM T88547 C5KGS0 10041278 Ki = 310 nM T88547 CY6HM5 10041770 Ki = 12.83 nM T88547 CM3L5T 10041887 Ki = 4 nM T88547 C3RPO9 10042466 Ki = 8 nM T88547 CCK0P4 10042708 Ki = 2.89 nM T88547 CIBU84 10043468 Ki = 1.9 nM T88547 CJ3V7G 10045023 Ki = 26 nM T88547 CZGN76 10048702 Ki = 335 nM T88547 C9B8JP 10049124 Ki = 16 nM T88547 C4T1PW 10061124 Ki = 21.66 nM T88547 CE4GX6 10064346 IC50 = 2740 nM T88547 CP0K9A 10064484 Ki = 1.54 nM T88547 C6V0IR 10064992 Ki = 4.34 nM T88547 C8FLO9 10065022 Ki = 440 nM T88547 CDX32I 10065362 Ki = 1.53 nM T88547 CP1S7J 10066063 Ki = 26.6 nM T88547 COZU58 10066419 Ki = 7 nM T88547 C0ISR6 10067170 Ki = 15 nM T88547 CU18XB 10069224 Ki = 25 nM T88547 CO69FB 10069973 Ki = 4295 nM T88547 C24TYX 10070045 IC50 = 92.8 nM T88547 CG5B2A 10070289 IC50 = 138 nM T88547 CQV2B9 10074800 Ki = 1.44 nM T88547 CI3D4F 10085466 Ki = 1.48 nM T88547 CI3R6W 10085970 Ki = 8.9 nM T88547 CROI43 10086447 Ki = 167 nM T88547 C9ECP3 10086666 Ki = 2.17 nM T88547 C9DX0V 10087782 Ki = 12 nM T88547 CVG5X1 10087999 Ki = 54 nM T88547 CIMQ96 10090127 Ki = 13 nM T88547 CKO26X 10090269 IC50 = 125 nM T88547 CU70GB 10090882 IC50 = 2100 nM T88547 CS3W1Z 10091077 Ki = 62.8 nM T88547 C7O8VH 10092041 IC50 = 64.1 nM T88547 CV48RC 10094571 Ki = 0.27 nM T88547 C0B8NJ 10094793 IC50 = 62 nM T88547 C1US0Q 10106826 Ki = 1.35 nM T88547 CRM6E0 10107042 Ki = 1.3 nM T88547 CM09JQ 10107360 Ki = 62.06 nM T88547 C6A5MJ 10107472 Ki = 243 nM T88547 CN4PY7 10108342 IC50 = 29 nM T88547 CQCN30 10108347 Ki = 26.7 nM T88547 CYKX67 10149140 Ki = 117 nM T88547 CTQ2A6 10176973 IC50 = 10.96 nM T88547 CZKG96 10200496 Ki = 3.4 nM T88547 C8R2AC 10243335 IC50 = 43 nM T88547 C51YTO 10243428 Ki = 7280 nM T88547 C31ZJX 10243991 IC50 = 1070 nM T88547 CKLA98 10246015 Ki = 410 nM T88547 C0NT8I 10248163 IC50 = 99.1 nM T88547 C0E5SL 10248164 IC50 = 246 nM T88547 C0UQ6P 10250792 IC50 = 53.5 nM T88547 CY9KM2 10250837 Ki = 1.02 nM T88547 CR4C1F 10253032 Ki = 5160 nM T88547 C6JH3D 10254219 Ki = 227 nM T88547 C4TK2U 10263215 Ki = 1042 nM T88547 CD5GU8 10263742 Ki = 1130 nM T88547 CWC2I4 10264753 Ki = 2.17 nM T88547 C48VLE 10264983 Ki = 6.6 nM T88547 CQJZ52 10264992 Ki = 1.18 nM T88547 CI29SE 10265752 Ki = 0.5 nM T88547 C1OER8 10266406 Ki = 21.3 nM T88547 C2F4ON 10266413 Ki = 0.69 nM T88547 CWF4D9 10267592 Ki = 710 nM T88547 CCP61G 10267880 IC50 = 7250 nM T88547 CW6UR5 10271046 IC50 = 234 nM T88547 C36PLT 10313891 Ki = 4 nM T88547 CP3Q4V 10314247 Ki = 1.45 nM T88547 CU3AC0 10314788 Ki = 10 nM T88547 CZM6T1 10316192 Ki = 11 nM T88547 CQZV80 10316321 Ki = 2.5 nM T88547 C7Q9KA 10319121 Ki = 0.51 nM T88547 C59KRL 10319931 Ki = 0.61 nM T88547 CNW60B 10331008 Ki = 83 nM T88547 CZ7AR2 10331473 Ki = 0.48 nM T88547 C34EYX 10333740 Ki = 0.96 nM T88547 C4K9SA 10334147 Ki = 21 nM T88547 CMX6Y0 10334410 Ki = 13 nM T88547 CARB42 10335164 Ki = 0.34 nM T88547 CT41RK 10336644 Ki = 9.6 nM T88547 C70MLB 10337045 Ki = 3 nM T88547 C5OT2E 10337119 Ki = 512.86 nM T88547 C60KJG 10337232 Ki = 265 nM T88547 CZI96H 10338172 Ki = 0.72 nM T88547 C3YCB5 10339444 Ki = 20.5 nM T88547 C2OCU0 10339767 Ki = 3 nM T88547 C9LKM0 10340180 IC50 = 7930 nM T88547 CO7C5M 10341072 Ki = 1.3 nM T88547 CF2U7Y 10342248 Ki = 2.78 nM T88547 C8KX0R 10342773 IC50 = 87.5 nM T88547 CF6NS0 10342845 Ki = 1.21 nM T88547 CS6P0J 10344430 Ki = 372 nM T88547 C52ZML 10354750 Ki = 6 nM T88547 CUK08H 10356159 Ki = 4.3 nM T88547 CZ9MG4 10356384 Ki > 100 nM T88547 CLG82T 10356463 Ki = 153 nM T88547 CN8PA7 10357986 Ki = 1.14 nM T88547 C6ZN0S 10358634 IC50 = 2640 nM T88547 CUD17B 10358719 Ki = 0.09 nM T88547 CG9WL5 10361439 IC50 = 198 nM T88547 C50OXW 10361564 Ki = 5 nM T88547 CW65RM 10365559 Ki = 27.22 nM T88547 CV2IT8 10365874 Ki = 1.3 nM T88547 C4I9US 10367771 Ki = 386.37 nM T88547 CM64TP 10368819 Ki = 22.8 nM T88547 CVY37K 10369311 Ki = 6 nM T88547 CWX81D 10369315 Ki = 0.88 nM T88547 CAYV90 10376919 Ki = 7.4 nM T88547 C9AJ7X 10378304 IC50 = 8 nM T88547 CO8NE3 10378306 IC50 = 1410 nM T88547 C2H1OB 10380647 Ki = 0.5 nM T88547 C7G9TF 10382446 Ki = 9 nM T88547 CYZN57 10383371 Ki = 2.19 nM T88547 CON6G8 10384067 IC50 = 55 nM T88547 CCZ74R 10384372 Ki = 9 nM T88547 CLY48W 10385977 IC50 = 59.9 nM T88547 C76DIU 10389641 IC50 = 707 nM T88547 C4DZ0M 10392655 Ki = 809 nM T88547 C34TLK 10402464 Ki = 1.34 nM T88547 C5SGY8 10404406 Ki = 13.4 nM T88547 C58RMD 10405079 Ki = 2.37 nM T88547 CHK46F 10405640 Ki = 101.7 nM T88547 CO34LY 10405821 IC50 = 8480 nM T88547 CDI85V 10406366 IC50 = 173 nM T88547 C5J6ZM 10407855 IC50 = 40 nM T88547 CKWY76 10408160 Ki = 0.5 nM T88547 CB67IL 10410177 Ki = 1.51 nM T88547 CZR8Q9 10422239 Ki = 5.4 nM T88547 CX1FR6 10423970 Ki = 26 nM T88547 C3JZ5Y 10426298 Ki = 16.76 nM T88547 CEKH47 10426373 Ki = 27 nM T88547 CLE64B 10426722 IC50 = 343 nM T88547 C2ZOF1 10428881 Ki = 46.98 nM T88547 CG0QM1 10429420 Ki = 24 nM T88547 C1A8XG 10430305 Ki = 19 nM T88547 CA1FD2 10430685 Ki = 61 nM T88547 C8Q4BP 10432985 Ki = 929.72 nM T88547 CN62ZX 10436105 Ki = 283 nM T88547 C1ZB7H 10446096 IC50 = 75 nM T88547 CO3EC1 10446949 IC50 = 13000 nM T88547 C36NJX 10447715 IC50 = 91 nM T88547 CBNM05 10447949 IC50 = 60 nM T88547 CS6E1O 10448420 Ki = 580 nM T88547 CYW8U4 10448771 Ki = 2.08 nM T88547 CMFL03 10449500 Ki = 9.4 nM T88547 CF25ZL 10449555 Ki = 2.66 nM T88547 CI0N2R 10449738 Ki = 11 nM T88547 CCP2O7 10450158 Ki = 3.6 nM T88547 C2G0AH 10450758 Ki = 35 nM T88547 C78IQN 10451373 Ki = 1066 nM T88547 CLY07Z 10453320 IC50 = 151 nM T88547 CACD15 10453690 IC50 = 11000 nM T88547 CAM7K8 10458892 Ki = 12900 nM T88547 CM48KH 10466885 Ki = 4450 nM T88547 C10HGT 10467460 Ki = 11.4 nM T88547 C6I2JZ 10467461 Ki = 4.8 nM T88547 C1B0JC 10470687 Ki = 4.3 nM T88547 CLE8W0 10470688 Ki = 2.9 nM T88547 C3BSH7 10473287 Ki = 1.2 nM T88547 C7GEB0 10474042 IC50 = 67.5 nM T88547 CTB5N8 10474751 Ki = 3.95 nM T88547 C8KE2J 10475196 Ki = 37 nM T88547 CUE5J0 10475634 IC50 = 52.2 nM T88547 C9S0EG 10491108 IC50 = 42.8 nM T88547 CLQU72 10493098 IC50 = 20.6 nM T88547 CIK95Q 10496036 IC50 > 1000 nM T88547 COES83 10496045 IC50 = 28.5 nM T88547 CU3GS8 10496297 IC50 = 110 nM T88547 C23KXT 10497826 Ki = 1.54 nM T88547 CU49FK 10498073 Ki = 29.6 nM T88547 CDMT59 10498740 IC50 = 65 nM T88547 COE3F4 10499273 Ki = 43.4 nM T88547 CI3TV1 10501583 Ki = 1.32 nM T88547 C4ZK6D 10502049 IC50 = 1050 nM T88547 C69BVP 10503221 IC50 = 150 nM T88547 CG72YU 10503374 IC50 = 8.6 nM T88547 C6K4WF 10504449 IC50 > 1000 nM T88547 C5HOS1 10517426 IC50 = 71.8 nM T88547 C30UGV 10517496 Ki = 19.8 nM T88547 CC94RX 10518276 IC50 = 164 nM T88547 C25ZVH 10521200 Ki = 20 nM T88547 C5NJ9X 10522573 Ki = 0.63 nM T88547 CFE07M 10522765 IC50 = 10 nM T88547 C9SGF2 10522997 Ki = 7.9 nM T88547 C3ZE8F 10524644 Ki = 1500 nM T88547 CXLS06 10525997 Ki = 4 nM T88547 C8Q0AM 10539358 Ki = 181 nM T88547 C94PRD 10540231 IC50 = 15.9 nM T88547 C9QX7K 10540232 IC50 = 20 nM T88547 C7XG2K 10541325 IC50 = 43.5 nM T88547 CK1IJ0 10542038 Ki = 62.3 nM T88547 C9NU4M 10542799 IC50 = 36.5 nM T88547 CJ7CY6 10545203 IC50 = 8 nM T88547 CA4P0N 10546938 Ki = 7.6 nM T88547 CKD9N5 10546961 Ki = 18.4 nM T88547 C5EJ9T 10550623 Ki = 31 nM T88547 CQD6C8 10551026 Ki = 5.9 nM T88547 CK27CJ 10551210 IC50 = 180 nM T88547 CEP7J1 10551313 Ki = 57 nM T88547 CZT94B 10564492 Ki = 7.7 nM T88547 C2PIU7 10564493 Ki = 6.4 nM T88547 CACP09 10566716 IC50 = 11.8 nM T88547 CJRB30 10567286 Ki = 127 nM T88547 CUR2O0 10568910 Ki = 61.66 nM T88547 C6OJL3 10569632 Ki = 6.457 nM T88547 CE2AQ9 10570139 Ki = 5.3 nM T88547 CO8SK3 10571211 Ki = 32.1 nM T88547 CD80FJ 10571528 Ki = 86 nM T88547 C10GOH 10575209 IC50 = 78 nM T88547 C2FAG0 10582642 Ki = 1.2 nM T88547 C1JH4Y 10582670 Ki = 1.9 nM T88547 CT78EI 10587586 Ki = 30.3 nM T88547 COR05F 10587917 IC50 = 18.5 nM T88547 CLD91R 10589924 Ki = 5.012 nM T88547 C9YSV1 10592242 Ki = 3.43 nM T88547 CW1L0N 10593974 IC50 = 330 nM T88547 C2WKD7 10594382 Ki = 63.9 nM T88547 C30YWC 10595615 Ki = 0.18 nM T88547 CONJ90 10596136 Ki = 16.6 nM T88547 CTJ5P1 10598454 IC50 = 381 nM T88547 CQ2M1Y 10599447 Ki = 18 nM T88547 CX1TS7 10599695 IC50 = 79 nM T88547 C9L0WQ 10599798 IC50 = 230 nM T88547 C4N7QJ 10599997 Ki = 1.1 nM T88547 CBAY37 10614630 Ki = 628 nM T88547 CXA13I 10615294 IC50 = 156 nM T88547 CAES37 10615793 IC50 = 97 nM T88547 CIQX09 10616126 Ki = 2.45 nM T88547 CS81FH 10616210 IC50 = 160 nM T88547 C42HFS 10616657 Ki = 115 nM T88547 CJ8T3N 10616816 IC50 > 1000 nM T88547 CG2RS0 10616993 Ki = 10.5 nM T88547 C8EH7Y 10617417 Ki = 7.63 nM T88547 CAT71Z 10618129 Ki = 145 nM T88547 CR5PI7 10618199 IC50 = 170 nM T88547 CZW69I 10618791 Ki = 42.2 nM T88547 CGJ0K6 10618918 Ki = 110.4 nM T88547 CSH12T 10619110 Ki = 29 nM T88547 C05AEY 10619619 Ki = 469 nM T88547 C8EX2V 10619631 IC50 = 130 nM T88547 CX7Q1J 10621853 IC50 = 34 nM T88547 CRS76W 10622914 Ki = 3.2 nM T88547 C7DQP5 10632134 Ki = 14280 nM T88547 C0UM2L 10634649 IC50 = 10.8 nM T88547 CCH7P1 10635235 Ki = 15.7 nM T88547 CAYM59 10635279 Ki = 63 nM T88547 CUE1G6 10637326 Ki = 736 nM T88547 CXO8K0 10638488 IC50 = 69.9 nM T88547 CFS6L3 10639616 Ki = 338.84 nM T88547 CGJ1U0 10640585 IC50 = 39.3 nM T88547 CE4UO3 10641401 Ki = 137.7 nM T88547 CI7T6M 10641797 Ki = 2.6 nM T88547 CO6TF0 10642179 Ki = 23.8 nM T88547 C7AZL4 10642861 IC50 = 420 nM T88547 CS46DA 10644162 Ki = 28 nM T88547 C3AGQ5 10645614 Ki = 0.7 nM T88547 CIN2U8 10646068 IC50 = 170 nM T88547 C4X8HV 10650002 IC50 = 4001 nM T88547 C2PGB1 10660038 Ki = 177 nM T88547 CAI09V 10661409 Ki = 0.6166 nM T88547 CW1H2S 10662563 IC50 = 14.4 nM T88547 C9PR7I 10662728 Ki = 365 nM T88547 C4AU9T 10663237 Ki = 15.2 nM T88547 CY9AE7 10664642 Ki = 5.9 nM T88547 CNX7J5 10665130 Ki = 3.87 nM T88547 CM1V7L 10665131 Ki = 3.17 nM T88547 CFX47R 10666733 Ki = 352 nM T88547 C0RBZ3 10666808 IC50 = 12 nM T88547 CXLA63 10668517 IC50 = 9 nM T88547 C1GPV6 10669784 IC50 = 1.5 nM T88547 CYF30E 10683536 IC50 > 1000 nM T88547 C8WEA9 10684798 Ki > 877 nM T88547 CVJ8N5 10686220 IC50 = 13.3 nM T88547 CCI6W0 10686221 IC50 = 31.8 nM T88547 C6YEV8 10687454 IC50 = 67 nM T88547 CZ27AV 10687985 IC50 = 40 nM T88547 C3SA7L 10689336 Ki = 7.32 nM T88547 CNK7Q5 10689502 Ki = 27.1 nM T88547 CIO4J5 10691389 IC50 = 5.7 nM T88547 CG01CM 10691769 Ki = 0.32 nM T88547 CBUK71 10695744 IC50 > 1000 nM T88547 CI52BL 10696254 Ki = 16.7 nM T88547 CCWU31 10710332 IC50 = 34 nM T88547 C9A1WC 10710941 IC50 = 39 nM T88547 CREK17 10711065 Ki = 159 nM T88547 CK2Y9B 10711119 Ki = 18.8 nM T88547 C6PJ4G 10711455 IC50 = 241 nM T88547 C4RVY0 10712370 Ki = 1.4 nM T88547 CJI3R5 10712473 Ki = 4.21 nM T88547 CN8S0W 10713214 IC50 = 4.5 nM T88547 C4R9DJ 10713754 Ki = 5.8 nM T88547 C52DUN 10713756 Ki = 1.91 nM T88547 C1VT7F 10714699 Ki = 7 nM T88547 CQ7L4I 10715370 Ki = 6520 nM T88547 C4QS9B 10716035 Ki = 457.09 nM T88547 CL8E5M 10717134 Ki = 21.4 nM T88547 CX05VT 10718443 Ki = 3.11 nM T88547 CYL27S 10718492 Ki = 230 nM T88547 C6Q3JA 10719188 Ki = 400 nM T88547 CG4S2Q 10719189 Ki = 6.2 nM T88547 CZ0A1O 10732853 IC50 = 231 nM T88547 CC84XI 10733148 Ki = 72 nM T88547 C9PES2 10733647 Ki = 70.79 nM T88547 CHO52Y 10733648 Ki = 234.42 nM T88547 C3Q4UE 10735303 IC50 = 125 nM T88547 CPZ24W 10735925 Ki > 1000 nM T88547 C8ONT1 10736122 Ki = 3.08 nM T88547 C1QJ2F 10738317 Ki = 139 nM T88547 C8ZH2S 10738339 Ki = 7.28 nM T88547 CA0Y3H 10739649 Ki = 80 nM T88547 C7QLT2 10741325 Ki = 1.2 nM T88547 C6XW5K 10741970 Ki = 1.7 nM T88547 CQ3F5D 10742360 IC50 = 41 nM T88547 C4L9AI 10742465 IC50 = 38 nM T88547 C08PYV 10754756 IC50 = 27 nM T88547 CL15XF 10757227 Ki = 5.754 nM T88547 C62VKE 10758083 Ki = 0.8 nM T88547 CWXZ23 10759399 Ki = 152 nM T88547 C3IQ9W 10761018 Ki = 7.762 nM T88547 C2COG9 10761980 Ki = 6.761 nM T88547 CPV9U1 10762065 Ki = 9.84 nM T88547 CQ1X0J 10762119 Ki = 5.22 nM T88547 C19OPJ 10763386 Ki = 14.2 nM T88547 C25ECH 10764130 IC50 = 29 nM T88547 CV54GW 10766338 Ki = 59 nM T88547 C7BZV3 10766454 IC50 = 30 nM T88547 CYSB34 10779682 IC50 = 45.7 nM T88547 C3RZF4 10779812 Ki = 202 nM T88547 C6JQ7A 10780443 IC50 > 10000 nM T88547 CN6CQ0 10780604 Ki = 286 nM T88547 CO9GR7 10782120 IC50 = 0.5 nM T88547 CA8IP1 10782132 Ki = 89.13 nM T88547 CJ62FW 10782325 Ki = 25 nM T88547 CN5U4I 10783531 Ki = 41.6 nM T88547 CZ5AK0 10784078 Ki = 5.6 nM T88547 CTU4Z6 10784820 Ki = 175 nM T88547 C57DMC 10787011 IC50 = 9.5 nM T88547 C2NG9Q 10789481 Ki = 1.1 nM T88547 CVT79G 10789674 IC50 = 59 nM T88547 CWJ40X 10789833 Ki = 56 nM T88547 C61YUS 10789834 Ki = 5.6 nM T88547 CN3RH8 10790095 Ki = 12.7 nM T88547 CM5S6D 10802506 Ki = 17.3 nM T88547 CAK53D 10805765 IC50 = 64 nM T88547 CT91OQ 10805927 Ki = 286.5 nM T88547 C0ACQ9 10807028 Ki = 43.8 nM T88547 C6IYD4 10807270 Ki = 20.1 nM T88547 C3VRX8 10807460 Ki = 758.58 nM T88547 CX6U3K 10807863 Ki = 1.8 nM T88547 C8O3ZD 10809006 Ki = 3.1 nM T88547 C1CUE8 10809630 IC50 = 110 nM T88547 C85KYQ 10811587 IC50 = 13 nM T88547 C0J7BR 10811875 Ki = 48 nM T88547 C2TPA5 10814571 Ki = 124.7 nM T88547 C3W7CM 10827238 Ki = 270 nM T88547 C3UHC7 10828366 Ki = 571 nM T88547 CES36I 10829775 Ki = 470 nM T88547 CGR8P0 10829840 Ki = 110 nM T88547 CK92FA 10831286 Ki = 1.2 nM T88547 CD8JF2 10831724 IC50 = 8.5 nM T88547 C6WD3U 10833752 Ki = 4.97 nM T88547 CCFI42 10834075 Ki = 2.89 nM T88547 C6HC0N 10834172 Ki = 9.55 nM T88547 C76JVF 10835756 Ki = 3.6 nM T88547 CRF51E 10835977 Ki = 0.14 nM T88547 CN2P9X 10836067 Ki = 41.8 nM T88547 CV4U5D 10836428 Ki = 5.8 nM T88547 CIBE62 10841374 IC50 = 3640 nM T88547 CAR05H 10849098 Ki = 23.8 nM T88547 CM7E2C 10850173 Ki = 19.6 nM T88547 CS8DX0 10851124 Ki = 1850 nM T88547 CW0P3J 10852782 Ki = 7.4 nM T88547 CJ9IL3 10852997 IC50 = 10.3 nM T88547 C6MC4P 10859662 Ki = 12.6 nM T88547 C62RCN 10862129 Ki = 298.56 nM T88547 C72FGM 10870255 Ki = 248.36 nM T88547 CI20YO 10871797 Ki = 13.3 nM T88547 CT7MS4 10881675 Ki = 1.83 nM T88547 C43WZD 10883323 Ki = 87.05 nM T88547 CRI50E 10885636 IC50 = 702 nM T88547 C5Z0DE 10893870 Ki = 15.1 nM T88547 C4J3YU 10895188 Ki = 51.94 nM T88547 C78FGZ 10902342 Ki = 0.86 nM T88547 C52TBK 10902954 Ki = 298.47 nM T88547 C42LHP 10903339 Ki = 11.7 nM T88547 CX65PW 10907460 IC50 = 482 nM T88547 C4SBO9 10915140 Ki = 2.07 nM T88547 C4L9XY 10924765 Ki = 12 nM T88547 CXO09C 10925078 Ki = 7.2 nM T88547 C8HG0I 10926436 Ki = 61.77 nM T88547 C1T9ZG 10936043 Ki = 2.21 nM T88547 CJA61X 10936501 Ki = 15.9 nM T88547 CA8NR0 10936584 Ki = 55.1 nM T88547 CN4TU6 10937393 Ki = 170 nM T88547 C7ACH1 10946809 Ki = 235.5 nM T88547 C9CEG5 10947083 Ki = 2.69 nM T88547 CB2E6K 10948128 Ki = 8.95 nM T88547 CYS1M8 10948383 IC50 = 158 nM T88547 CO04EB 10948807 Ki = 141.36 nM T88547 CP0J7O 10950137 Ki = 346.9 nM T88547 CBQ2J3 10969171 Ki = 1.4 nM T88547 CZ61YN 10969173 Ki = 1.7 nM T88547 CYB4W9 10969339 Ki = 31.25 nM T88547 C9QBS4 10970390 Ki = 4.64 nM T88547 C5LZH9 10980649 Ki = 6.64 nM T88547 CQ7A1S 10981062 Ki = 3.97 nM T88547 CE5K8F 10991643 Ki = 10.9 nM T88547 C7R1CB 11001837 Ki = 7.27 nM T88547 C0UY4P 11003384 Ki = 183 nM T88547 CJT8Y7 11012319 Ki = 269.15 nM T88547 CJ78DG 11013161 Ki = 12.4 nM T88547 C6YWX4 11013162 Ki = 12.7 nM T88547 CE04WV 11016132 Ki = 2.31 nM T88547 C82RNS 11016707 Ki = 3.49 nM T88547 CQ6M1S 11028157 Ki = 751 nM T88547 CGA2C4 11034660 Ki = 43.7 nM T88547 C89XHJ 11034920 Ki = 1390 nM T88547 C8SH3D 11035595 Ki = 19.07 nM T88547 CB7N1P 11035765 IC50 = 328 nM T88547 CXPD18 11045363 Ki = 1.09 nM T88547 C4LE3O 11046757 Ki = 9.33 nM T88547 C23JHR 11047568 IC50 = 2170 nM T88547 CS9FX5 11064325 Ki = 19800 nM T88547 CGI1R9 11091108 Ki = 13.1 nM T88547 CK2WT1 11102433 Ki = 4.29 nM T88547 CU21VJ 11109490 Ki = 2.18 nM T88547 CF3D0J 11109952 Ki = 2.16 nM T88547 C2MR9D 11110106 Ki = 7.16 nM T88547 CF29UZ 11111624 Ki = 125.41 nM T88547 C65WYU 11120436 Ki = 5.66 nM T88547 CY2N6C 11142430 Ki = 149.84 nM T88547 C49ECI 11143217 Ki = 1.87 nM T88547 C1BIZ9 11143323 Ki = 7.24 nM T88547 CU6PV0 11143820 IC50 = 581 nM T88547 C74YMR 11152920 Ki = 5.54 nM T88547 CYS2X0 11154079 Ki = 1.2 nM T88547 CC1AT3 11165837 Ki = 3078 nM T88547 CMA72C 11168272 Ki = 18 nM T88547 C8SL0F 11189143 Ki = 16.2 nM T88547 CU5ND9 11191741 Ki = 1159 nM T88547 CQ9NP6 11198145 Ki = 2 nM T88547 CK34VH 11199981 Ki = 1.54 nM T88547 CAZ9K5 11233111 Ki = 0.61 nM T88547 C27PSA 11234042 Ki = 3.38 nM T88547 C0UMB4 11234470 Ki = 36.4 nM T88547 CM59CS 11235994 Ki = 15.1 nM T88547 C3NF5Z 11237443 Ki = 15.4 nM T88547 CZKE17 11268724 Ki = 0.36 nM T88547 CUSN36 11281378 Ki = 3.07 nM T88547 CZS56H 11292472 Ki = 1.52 nM T88547 CQ0FP3 11292970 Ki = 10000 nM T88547 CGZM12 11302686 Ki = 0.036 nM T88547 CQ29OL 11303155 Ki = 1.45 nM T88547 CQ2Z6J 11304676 Ki = 276.5 nM T88547 CBAU26 11315257 Ki = 21.8 nM T88547 C0LVZ4 11317999 Ki = 189.1 nM T88547 CJT02X 11326158 Ki = 28.7 nM T88547 CTIX74 11338096 Ki = 10400 nM T88547 C3JBI0 11338418 Ki = 0.3 nM T88547 CL7O2I 11349674 Ki = 9.4 nM T88547 CENY72 11360254 Ki > 1000 nM T88547 CY20HV 11372576 Ki = 9.9 nM T88547 CN96RT 11381875 Ki = 0.4 nM T88547 C3V7NH 11405584 Ki = 1.5 nM T88547 C17XGQ 11405620 Ki = 1.57 nM T88547 CGH8L0 11405872 Ki = 2.4 nM T88547 C6WM2A 11406043 Ki = 1.4 nM T88547 CMI90K 11407131 Ki = 0.3 nM T88547 C7CX1Z 11407133 Ki = 0.4 nM T88547 C4HVO6 11416825 Ki = 0.22 nM T88547 CGA4V6 11428574 Ki = 1.57 nM T88547 CGU24X 11428679 Ki = 2.45 nM T88547 C7GB8T 11439301 Ki = 0.31 nM T88547 C2B9FV 11440556 Ki = 36.3 nM T88547 CJW6P0 11451147 Ki = 0.69 nM T88547 C6GXJ4 11451971 Ki = 11.9 nM T88547 CL61VY 11462448 Ki = 5.4 nM T88547 CAL0Z7 11488451 Ki = 2932 nM T88547 CVU67H 11494142 Ki = 17.2 nM T88547 CUTX86 11494380 Ki = 6.9 nM T88547 CQX19K 11501260 Ki = 10.4 nM T88547 C0KBI1 11501613 Ki = 8.2 nM T88547 CN0OV4 11508643 Ki = 5.5 nM T88547 CCQ5N8 11518209 Ki = 26 nM T88547 C5MRO3 11522946 Ki = 5.2 nM T88547 CN35YZ 11531125 Ki = 10.2 nM T88547 CBFZ60 11531451 Ki = 4 nM T88547 C0HL2V 11531518 Ki = 24 nM T88547 CWXL39 11532920 Ki = 16 nM T88547 CB6PI4 11537339 Ki = 10 nM T88547 CVUI98 11544226 Ki > 1000 nM T88547 CU3Z9X 11544597 Ki = 294 nM T88547 C5TZV9 11552718 Ki = 13.3 nM T88547 CY1H3V 11558654 IC50 = 15.5 nM T88547 C26EIT 11567446 Ki = 9.9 nM T88547 COPG87 11573361 Ki = 7 nM T88547 C3UQL8 11573971 Ki = 10.8 nM T88547 CFT29G 11594918 Ki = 9.9 nM T88547 C65ESO 11602582 Ki = 9.9 nM T88547 C9XM1Q 11604103 Ki = 224 nM T88547 C0TAC4 11610271 Ki = 854 nM T88547 C51DOW 11617627 Ki = 17.6 nM T88547 CUCN59 11618199 Ki = 741 nM T88547 C8IE7O 11624298 Ki = 8.2 nM T88547 CPA75G 11625126 Ki = 7.1 nM T88547 CO19EP 11632093 Ki = 11.7 nM T88547 CW42YV 11646372 Ki = 11.1 nM T88547 CES7K4 11652595 IC50 = 11.3 nM T88547 C8B5GK 11652762 Ki = 15.7 nM T88547 C1HDM5 11653679 Ki = 23.44 nM T88547 C8EHT5 11659822 Ki = 47 nM T88547 CFB42T 11667265 Ki = 16.7 nM T88547 CO23PC 11668112 Ki = 172 nM T88547 CN0TZ2 11682186 Ki = 9.4 nM T88547 C3XDB2 11704592 Ki = 44 nM T88547 CF02CY 11704696 Ki > 1000 nM T88547 CWM71X 11718233 Ki = 14.8 nM T88547 C3KU0D 11722772 Ki = 0.49 nM T88547 C6ZGX3 11723852 Ki = 0.97 nM T88547 CME0R3 11725031 Ki = 2 nM T88547 CX1ZF4 11725919 Ki = 29.9 nM T88547 CD9V5B 11733099 Ki = 15.41 nM T88547 CWX41Z 11739209 Ki = 2.16 nM T88547 CDFB43 11743300 Ki = 26700 nM T88547 C1U6PW 11748820 Ki = 29.3 nM T88547 C9GNC5 11758674 Ki = 10100 nM T88547 CBY2Q9 11760579 Ki > 1000 nM T88547 CZ8E3X 11771731 Ki = 125 nM T88547 CDW1T8 11776562 Ki = 28.7 nM T88547 CFSU16 11777643 IC50 = 341 nM T88547 C8DVY0 11777930 Ki = 10 nM T88547 C0P3JO 11782688 Ki = 5.83 nM T88547 CEM4V0 11783308 Ki = 23.88 nM T88547 CJ5Z9H 11784333 Ki = 95.3 nM T88547 CW5L6Q 11791714 Ki = 5.8 nM T88547 C9QI0E 11791902 Ki = 66 nM T88547 CZUE50 11792320 Ki = 54 nM T88547 C6ZQF2 11792374 Ki = 4.56 nM T88547 CWE12Y 11792375 Ki = 18 nM T88547 CZH6S4 11793400 Ki = 121 nM T88547 C3D4PU 11793930 Ki = 8.7 nM T88547 CH6B0Y 11793931 Ki = 3.92 nM T88547 CYR0V7 11794387 IC50 > 1000 nM T88547 C6U2RY 11796923 Ki = 2.5 nM T88547 C9C7HV 11797295 IC50 = 43 nM T88547 C4X8UL 11800052 Ki = 121.8 nM T88547 CHOE91 11808864 Ki = 1.81 nM T88547 CZQ51Y 11810652 Ki = 10.2 nM T88547 CN9M8E 11811722 IC50 = 1250 nM T88547 CT1L3N 11822555 Ki = 7.33 nM T88547 CH91AX 11824300 Ki = 148 nM T88547 CXLW54 11948707 Ki = 180 nM T88547 CT8Q2B 11957591 IC50 = 3.802 nM T88547 CN82RK 11957597 Ki = 118 nM T88547 CKG40P 12084044 Ki = 121 nM T88547 C3ZC4D 12084050 Ki = 69 nM T88547 CCA4D0 12084052 Ki = 96 nM T88547 C6NCO1 12084053 Ki = 28 nM T88547 CE7ZN1 12084054 Ki = 6.2 nM T88547 C6DQ4H 12084055 Ki = 23.4 nM T88547 CZ14EL 12084056 Ki = 375 nM T88547 C5HS8Q 12259685 Ki = 1.7 nM T88547 CSQ2J7 12329382 Ki = 660 nM T88547 C2FOU9 12347284 Ki = 11.7 nM T88547 CA45VN 12351937 Ki = 664 nM T88547 CS5IZ8 12371110 Ki = 6750 nM T88547 CSY9N8 12371111 Ki = 2733 nM T88547 C3Y9UN 12491976 IC50 = 338.84 nM T88547 CQ9F1W 12491977 IC50 = 446.68 nM T88547 C3E7QH 12628908 IC50 = 4100 nM T88547 C2GH7O 12730763 Ki = 20 nM T88547 C4G0MK 12730765 Ki = 29 nM T88547 CH81JK 12730766 Ki = 29 nM T88547 C3H1AN 12874567 Ki = 13.6 nM T88547 CL6G8E 12874569 Ki = 31 nM T88547 CBK95L 12914591 Ki = 48.2 nM T88547 C6LV2S 13011906 Ki = 10.8 nM T88547 C23ELH 13078350 IC50 = 6605 nM T88547 CCG14E 13091356 Ki = 165.96 nM T88547 CYN95Z 13091359 Ki = 81 nM T88547 CYV6B5 13781931 IC50 = 13.8 nM T88547 C2SEG3 13781932 IC50 = 66 nM T88547 CG08MN 13781936 IC50 = 65 nM T88547 C3FCB2 13781939 IC50 = 356 nM T88547 CL7XE8 13998486 Ki = 6 nM T88547 C7VG5C 14040442 IC50 = 1516 nM T88547 CX20PD 14125583 IC50 = 32 nM T88547 CS61DC 14291221 Ki = 418 nM T88547 CJNM56 14292033 IC50 = 220 nM T88547 CC8A3Q 14368937 Ki = 21 nM T88547 CQ9G0L 14368954 Ki = 7 nM T88547 CIE32U 14368960 Ki = 12 nM T88547 CYW76P 14742527 Ki > 1000 nM T88547 C50XLA 14771399 IC50 = 2593 nM T88547 CXM7W9 14771402 IC50 = 418 nM T88547 CA4OM8 14771405 IC50 = 2100 nM T88547 CV87AM 14771416 IC50 = 6058 nM T88547 CNMV48 14771443 IC50 = 77 nM T88547 CDG54I 14771450 Ki = 11 nM T88547 C91VRA 14771452 Ki = 8.66 nM T88547 CHPJ17 14771454 Ki = 1372 nM T88547 CUXT02 14771457 Ki = 456 nM T88547 CA2LP1 14771459 Ki = 7212 nM T88547 C8X7UK 14771468 IC50 = 966 nM T88547 C17WBC 14771473 IC50 = 125 nM T88547 CL7PU3 14771475 IC50 = 37 nM T88547 C6EUR2 14771480 Ki = 89.5 nM T88547 CTAB86 14771482 Ki = 30.5 nM T88547 CRJ0L3 14771666 IC50 = 96 nM T88547 CE0KP4 14771667 IC50 = 59 nM T88547 CM29BA 14771668 IC50 = 36 nM T88547 C5SU1R 14771669 IC50 = 125 nM T88547 CWMO41 14771670 IC50 = 215 nM T88547 CPB79U 14771672 IC50 = 33 nM T88547 C7M1AK 14771673 IC50 = 8110 nM T88547 CTBR56 14771675 IC50 = 203 nM T88547 CQ1ZC3 14771677 IC50 = 16 nM T88547 CX4H7W 14771682 IC50 = 750 nM T88547 CIY37H 14771684 IC50 = 21 nM T88547 CP4LQ5 14771685 IC50 = 37 nM T88547 CR67MN 14771686 IC50 = 42 nM T88547 CEQV06 14771688 IC50 = 440 nM T88547 CH2R4M 14771689 IC50 = 850 nM T88547 CDHN24 14771691 IC50 = 920 nM T88547 C3WK2C 14771692 IC50 = 935 nM T88547 CJ21YE 14771693 IC50 = 1200 nM T88547 CJY5N0 14771694 IC50 = 12 nM T88547 C2NW9K 14771695 IC50 = 6 nM T88547 C47EWB 14771696 IC50 = 8 nM T88547 CF6OB9 14771697 IC50 = 20 nM T88547 CRK3S4 14771698 IC50 = 300 nM T88547 CO4Z3M 14771699 IC50 = 4 nM T88547 C6A4YT 14771702 IC50 = 6 nM T88547 CS9Z3L 14771705 IC50 = 25 nM T88547 C8S0BC 14771707 IC50 = 155 nM T88547 CU94AL 14771709 IC50 = 5.2 nM T88547 C2FO3S 14771711 IC50 = 15 nM T88547 CF2L5J 14771713 IC50 = 16 nM T88547 CL0GD1 14771715 IC50 = 112 nM T88547 C8B9LE 14771717 IC50 = 245 nM T88547 CGJB25 14771719 IC50 = 345 nM T88547 C6JM8H 14771721 IC50 = 370 nM T88547 C0BZJ6 14771723 IC50 = 970 nM T88547 CCW53V 14771725 IC50 = 18 nM T88547 CCMA03 14771728 IC50 = 118 nM T88547 CXGT50 14771729 IC50 = 962 nM T88547 CZSE76 14771731 IC50 = 5100 nM T88547 CCZ3L7 14771734 IC50 = 237 nM T88547 CL7NO6 14771736 IC50 = 238 nM T88547 C64VXZ 14771738 IC50 = 8 nM T88547 CQ92IT 14771742 IC50 = 21.1 nM T88547 C53BMJ 14771744 IC50 > 10000 nM T88547 CDP91Q 14831233 Ki = 9.3 nM T88547 CX7YM2 14831240 Ki = 2.6 nM T88547 CYA34X 14831246 Ki = 97 nM T88547 CXBP45 14831249 Ki = 56 nM T88547 C6CR4J 14895995 IC50 = 10 nM T88547 C42OVT 14941803 Ki = 16.6 nM T88547 C0AY3O 14952694 Ki = 125 nM T88547 CI6MH4 14970526 IC50 = 8 nM T88547 C83VFC 14970527 IC50 = 500 nM T88547 C3MG6W 14970528 IC50 = 100 nM T88547 CKRQ36 14970529 IC50 = 495 nM T88547 C1AYO7 14970530 IC50 = 235 nM T88547 CNF3X6 14970531 IC50 = 400 nM T88547 CA1QS4 14970532 IC50 = 281 nM T88547 C6PO3M 14970533 IC50 = 158 nM T88547 CQ3YR9 14970534 IC50 = 105 nM T88547 CP4G5R 14970535 IC50 = 23 nM T88547 CP6FW7 14970536 IC50 = 25 nM T88547 C6IZC7 14970537 IC50 = 66 nM T88547 CLYJ93 14970538 IC50 = 7 nM T88547 C25QOE 14976641 Ki = 4400 nM T88547 C46ZRG 14977560 IC50 = 140 nM T88547 C3XV5J 14982949 IC50 = 40 nM T88547 CPBC12 14982950 IC50 = 257 nM T88547 CSX4B6 14982951 IC50 = 720 nM T88547 C2SE6U 14982952 IC50 = 1800 nM T88547 CY3FM7 14982953 IC50 = 432 nM T88547 CC2HP8 14982954 IC50 = 165 nM T88547 CR8ZX1 14982955 IC50 = 227 nM T88547 CIG1W9 14982956 IC50 = 202 nM T88547 CNB0U1 14982957 IC50 = 297 nM T88547 CLG2A3 14982961 IC50 = 77 nM T88547 C83QWH 14982964 IC50 = 88 nM T88547 CJU87A 14982965 IC50 = 54 nM T88547 CJ2PE3 14982966 IC50 = 24 nM T88547 CY82JH 14982968 IC50 = 23 nM T88547 C59ETV 14982969 IC50 = 52 nM T88547 C8FHX4 14982970 IC50 = 100 nM T88547 CQV51D 14982971 IC50 = 237 nM T88547 CIFL16 14982976 IC50 = 80 nM T88547 CGE08Y 14982977 IC50 = 226 nM T88547 CR72BK 14982978 IC50 = 155 nM T88547 CIJ47C 14982979 IC50 = 164 nM T88547 COC5A3 14982980 IC50 = 53 nM T88547 C1Y4DM 14982981 IC50 = 1900 nM T88547 CODB98 14982982 IC50 = 49 nM T88547 C1Z9BL 14982983 IC50 = 347 nM T88547 CRF43C 14982984 IC50 = 2100 nM T88547 C3CXH1 14982992 IC50 = 33 nM T88547 C3BK0M 14982993 IC50 = 92 nM T88547 C0YQF8 14982994 IC50 = 45 nM T88547 C31OGY 14982995 IC50 = 16 nM T88547 CELY61 14982996 IC50 = 22 nM T88547 CU8X7Q 14982997 IC50 = 36 nM T88547 C89ZMJ 14983027 IC50 = 29 nM T88547 CJB9L5 14983028 IC50 = 119 nM T88547 CE2LO0 14983029 IC50 = 175 nM T88547 C7V0FZ 14983030 IC50 = 129 nM T88547 C8XK3F 14983031 IC50 = 320 nM T88547 C0F2YM 14983032 IC50 = 76 nM T88547 COHF72 14983033 IC50 = 194 nM T88547 CE62QX 14983034 IC50 = 164 nM T88547 C9XB8N 14983035 IC50 = 95 nM T88547 CT9B0C 14983036 IC50 = 493 nM T88547 CUD3A8 14983037 IC50 = 254 nM T88547 CE0OG6 14983038 IC50 = 159 nM T88547 CL0QW6 14983039 IC50 = 50 nM T88547 CV4XG6 14983040 IC50 = 51 nM T88547 CAD38J 14983041 IC50 = 190 nM T88547 C83IQA 14983042 IC50 = 46 nM T88547 CHMC30 14983043 IC50 = 84 nM T88547 C0E1GY 14983044 IC50 = 139 nM T88547 CG7SN0 14983045 IC50 = 95 nM T88547 CE2XK1 14983046 IC50 = 32 nM T88547 CW3R4M 14983047 IC50 = 63 nM T88547 C5YAV6 14983048 IC50 = 73 nM T88547 CY40QK 14983049 IC50 = 119 nM T88547 CMPN17 14983050 IC50 = 67 nM T88547 CHG9L5 14983053 IC50 = 34 nM T88547 CI79PE 14983054 IC50 = 26 nM T88547 CY1ZT7 14983055 IC50 = 93 nM T88547 C4X9RT 15034720 Ki = 41 nM T88547 C0JVK6 15034721 Ki = 34 nM T88547 C6FLJ0 15034722 Ki = 14 nM T88547 C1XUR9 15034723 Ki = 15 nM T88547 CYJ8D3 15034724 Ki = 19 nM T88547 C1E9DR 15034725 Ki = 18 nM T88547 C0CML8 15034727 Ki = 16 nM T88547 CRD98J 15034728 Ki = 62 nM T88547 CW97AB 15034729 Ki = 31 nM T88547 C7DE2A 15034730 Ki = 17 nM T88547 C0XTN3 15034731 Ki = 5 nM T88547 CU3V1E 15034733 Ki = 16 nM T88547 C3DIU6 15034734 Ki = 3 nM T88547 CF6BC5 15034735 Ki = 24 nM T88547 CSZ6G9 15034737 Ki = 15 nM T88547 C20NWP 15034738 Ki = 2 nM T88547 CU5I8Q 15034740 Ki = 250 nM T88547 CT91RK 15034743 Ki = 170 nM T88547 CGA52B 15034744 Ki = 19 nM T88547 CFQB36 15061885 Ki = 9.5 nM T88547 COQ0S2 15061886 Ki = 6.2 nM T88547 CE74WO 15061887 Ki = 3.4 nM T88547 C4R7ZN 15061888 Ki = 9.3 nM T88547 CSI1G0 15061889 Ki = 6.3 nM T88547 CI8CY0 15061890 Ki = 27.4 nM T88547 C7NR1V 15061896 Ki = 27.1 nM T88547 CG3T6K 15061897 Ki = 6 nM T88547 C4S2OB 15061898 Ki = 8.8 nM T88547 C6BJ0T 15061899 Ki = 12 nM T88547 CV8K6X 15061903 Ki = 83.2 nM T88547 CO31ZL 15061905 Ki = 7.9 nM T88547 CY1KZ4 15061906 Ki = 20 nM T88547 C6NL4F 15065448 IC50 = 17 nM T88547 C7R4WQ 15065449 IC50 = 7 nM T88547 C82EDI 15065450 IC50 = 7 nM T88547 CX7DC9 15065451 IC50 = 8 nM T88547 C61DXO 15065452 IC50 = 13 nM T88547 CYTG20 15065453 IC50 = 9 nM T88547 COBY80 15065454 IC50 = 3.2 nM T88547 CE35OQ 15065456 IC50 = 8 nM T88547 CAK96V 15113293 Ki = 1.76 nM T88547 CAL9M2 15113300 Ki = 5.78 nM T88547 C4H1NE 15113301 Ki = 277 nM T88547 CU7I0M 15113304 Ki = 1.35 nM T88547 COD14I 15113305 Ki = 11.7 nM T88547 CC4U7N 15113306 Ki = 0.84 nM T88547 CZ5XG0 15113307 Ki = 2.09 nM T88547 CQ26WU 15113308 Ki = 0.73 nM T88547 CN75UR 15113309 Ki = 20.18 nM T88547 CJO12C 15113311 Ki = 1.46 nM T88547 C8L6WJ 15113312 Ki = 0.62 nM T88547 C0BUH8 15113313 Ki = 0.38 nM T88547 CP7Z9O 15149381 IC50 = 116 nM T88547 C7ZQ8S 15149384 IC50 = 1612 nM T88547 C3ZK6U 15149386 IC50 = 474 nM T88547 CGBZ29 15149390 IC50 = 3560 nM T88547 CPZ2Q5 15149391 IC50 = 1276 nM T88547 CA10MG 15149392 IC50 = 1763 nM T88547 CR6HS1 15149393 IC50 = 2750 nM T88547 CZTR71 15149394 IC50 = 234 nM T88547 CR19PC 15149395 IC50 = 81 nM T88547 CK6CR7 15149396 IC50 = 348 nM T88547 CV5WQ2 15149397 IC50 = 534 nM T88547 CD1G7K 15149398 IC50 = 4876 nM T88547 CXB9C3 15149399 IC50 = 400 nM T88547 COK78H 15149400 IC50 = 262 nM T88547 C2NW3G 15149401 IC50 = 148 nM T88547 C8UCG2 15149402 IC50 = 88 nM T88547 C7KA2N 15149403 IC50 = 21 nM T88547 C1HR0I 15149404 IC50 = 105 nM T88547 C9KNO8 15149405 IC50 = 66 nM T88547 CW5MC6 15149406 IC50 = 129 nM T88547 CCH01D 15149407 IC50 = 133 nM T88547 CM2P4G 15149408 IC50 = 1483 nM T88547 CEWY20 15149409 IC50 = 702 nM T88547 CG7Q6W 15149411 IC50 = 1382 nM T88547 CX79WN 15149412 IC50 = 86 nM T88547 C6QL3P 15149413 IC50 = 3044 nM T88547 CHBC48 15149414 IC50 = 44 nM T88547 CN0P7T 15149415 IC50 = 8085 nM T88547 CAG3U8 15149416 IC50 = 836 nM T88547 CWN18O 15149417 IC50 = 85 nM T88547 CCH6M2 15149418 IC50 = 76 nM T88547 C8K5YO 15149419 IC50 = 231 nM T88547 CP83UL 15149420 IC50 = 267 nM T88547 C6O1FB 15149421 IC50 = 212 nM T88547 C7F1XV 15149422 IC50 = 482 nM T88547 CPE03W 15149426 IC50 = 3950 nM T88547 CV79PM 15163132 IC50 = 5.495 nM T88547 CG64QT 15163133 IC50 = 6.761 nM T88547 CSYU86 15163134 IC50 = 69.18 nM T88547 C20RCB 15163135 IC50 = 74.13 nM T88547 CM82BJ 15163136 IC50 = 6.761 nM T88547 CXWA38 15163138 IC50 = 4.786 nM T88547 CFMK89 15163140 IC50 = 1.047 nM T88547 CD4N5E 15163141 Ki = 0.6 nM T88547 C6JO1G 15163142 IC50 = 2.291 nM T88547 C4TX7I 15163143 IC50 = 2.884 nM T88547 CU3KS6 15163144 IC50 = 5.012 nM T88547 C8GZW1 15163145 IC50 = 6.607 nM T88547 CPIL08 15163146 IC50 = 10.23 nM T88547 CX3L5P 15163147 IC50 = 18.2 nM T88547 CI48UB 15163148 IC50 = 1.413 nM T88547 C9WFS6 15163149 IC50 = 1.66 nM T88547 CMZ73A 15163150 IC50 = 6.761 nM T88547 CTZ6J7 15163151 IC50 = 14.13 nM T88547 C1QZA4 15163152 IC50 = 9.55 nM T88547 C9V2LE 15163153 IC50 = 6.31 nM T88547 CEJ3H5 15163154 IC50 = 5.495 nM T88547 CAM8N1 15163155 IC50 = 11.22 nM T88547 C07FGX 15163160 IC50 = 1.349 nM T88547 C59BLX 15163161 IC50 = 1.514 nM T88547 C1JY2C 15163162 IC50 = 2.042 nM T88547 C36LSH 15163163 IC50 = 3.467 nM T88547 CGW2U3 15163164 IC50 = 3.162 nM T88547 CT0FG7 15163165 IC50 = 16.22 nM T88547 CKQL79 15166841 Ki = 2.72 nM T88547 CLIK54 15166843 Ki = 44.5 nM T88547 CL25QN 15166844 Ki = 10.3 nM T88547 CRX06M 15166845 Ki = 2.13 nM T88547 CA58OD 15175719 Ki = 1.19 nM T88547 C6EQD1 15175722 Ki = 0.54 nM T88547 CB0M5G 15205702 Ki = 46.5 nM T88547 C2B9YF 15205887 Ki = 1200 nM T88547 CX8YP7 15229597 Ki = 7 nM T88547 C4XSK7 15230909 IC50 = 100 nM T88547 CCZ8K3 15288693 Ki = 3 nM T88547 CWJ12B 15340879 Ki = 3 nM T88547 CR4UB7 15379806 IC50 = 26 nM T88547 CFQU06 15379808 IC50 = 16 nM T88547 CXP2Q0 15428989 Ki = 1.4 nM T88547 CZ72SA 15489265 Ki = 78.7 nM T88547 C65SCN 15599151 Ki = 484 nM T88547 CD0ZG3 15601069 Ki = 5200 nM T88547 CW3U0L 15646123 IC50 = 1212 nM T88547 C7UMB1 15646135 IC50 = 25 nM T88547 C0CXT6 15646139 IC50 = 37 nM T88547 C37SJN 15646141 IC50 = 38 nM T88547 CF2G1M 15646180 IC50 = 54 nM T88547 CRYD49 15657191 IC50 = 3305 nM T88547 C9P8QD 15657199 IC50 = 16.98 nM T88547 C1D0AP 15657202 IC50 = 0.2884 nM T88547 CSI49R 15657205 IC50 > 10000 nM T88547 C47CMD 15657207 IC50 = 10.47 nM T88547 C3E1TB 15657209 IC50 = 79.43 nM T88547 CUX59A 15657212 IC50 = 8.9 nM T88547 CG4LS3 15657214 IC50 = 117 nM T88547 C2F1JU 15657216 IC50 = 26.5 nM T88547 C12MGR 15657218 IC50 = 2.239 nM T88547 C5YG3C 15657219 IC50 = 3342 nM T88547 C57CUI 15701658 Ki = 146 nM T88547 CIUE86 15701660 Ki = 55.7 nM T88547 C4RX3J 15701661 Ki = 140 nM T88547 C1AYL6 15701662 Ki = 3.5 nM T88547 CU96AV 15701663 Ki = 3.1 nM T88547 CGEF49 15701664 Ki = 38 nM T88547 C1U5HG 15701665 Ki = 412 nM T88547 C1YFB9 15723883 Ki = 2.6 nM T88547 CDB0N6 15723885 Ki = 5.4 nM T88547 CVG95S 15723887 Ki = 2.8 nM T88547 CLN2V3 15723888 Ki = 125 nM T88547 C0JN7F 15723897 Ki = 4 nM T88547 CS98BY 15729885 IC50 = 23 nM T88547 C5NQL7 15729886 IC50 = 51 nM T88547 C6IFV4 15729897 IC50 = 1520 nM T88547 CU0J4B 15729898 IC50 > 45 nM T88547 C18DGR 15729900 IC50 = 12 nM T88547 C6ACS9 15729901 IC50 = 88 nM T88547 CJA86K 15729905 IC50 = 213 nM T88547 COLX61 15729907 IC50 = 504 nM T88547 CN95AB 15729914 IC50 = 227 nM T88547 CP7E8U 15729917 IC50 = 215 nM T88547 C7BH5E 15729921 IC50 > 1 nM T88547 CE87JV 15729922 IC50 = 3500 nM T88547 CG6FM7 15729925 IC50 > 2 nM T88547 C2LK6I 15729927 IC50 = 52 nM T88547 C7JK2U 15751758 IC50 = 3467.37 nM T88547 C9WX1R 15751761 IC50 = 1174.9 nM T88547 CE4TS7 15751762 IC50 = 338.84 nM T88547 C2CY5H 15751763 IC50 = 6.31 nM T88547 CMR8Q4 15751764 IC50 = 3.09 nM T88547 C40GZI 15751790 IC50 = 1.862 nM T88547 CZ69AV 15751791 IC50 = 3.981 nM T88547 C3QXB0 15751793 IC50 = 2.138 nM T88547 C4N9EK 15751794 IC50 = 1.413 nM T88547 CHL8I9 15767674 Ki = 1.57 nM T88547 C7JVH8 15767675 Ki = 82.5 nM T88547 CYCG42 15767676 Ki = 18.4 nM T88547 C45ITA 15767677 Ki = 5.68 nM T88547 C7H0OA 15767678 Ki = 1.47 nM T88547 CWH7G0 15767679 Ki = 1.75 nM T88547 CGF67P 15767680 Ki = 10.4 nM T88547 C7CLQ9 15767681 Ki = 3.81 nM T88547 CFH51J 15767682 Ki = 7.16 nM T88547 CR3LW7 15767683 Ki = 18.5 nM T88547 CFMC10 15767684 Ki = 130.6 nM T88547 CCP96Z 15767685 Ki = 4.68 nM T88547 CG8KR9 16005860 IC50 < 20 nM T88547 CAUP23 16048564 Ki = 2.2 nM T88547 C10CLM 16061352 Ki = 207 nM T88547 CTME96 16202156 Ki = 2150 nM T88547 CZ2IS9 16660294 Ki > 10000 nM T88547 CBH0C8 16664364 Ki = 2.1 nM T88547 CSNM61 16730082 Ki = 36.8 nM T88547 C0LEG4 17159068 Ki = 16 nM T88547 CA6E9Q 17159204 Ki = 2.5 nM T88547 C8O7EW 17176477 Ki = 15 nM T88547 C45JHX 17644936 Ki > 100 nM T88547 C7MST8 17758676 Ki = 3450 nM T88547 CM36GJ 17867053 Ki = 8 nM T88547 C21FJV 17867054 Ki = 5 nM T88547 CCM1L3 18118650 Ki = 10 nM T88547 CZ31UL 18118651 Ki = 37 nM T88547 C9UE6C 18118654 Ki = 40 nM T88547 C30VIU 18703006 Ki = 0.76 nM T88547 CD4BH5 18703016 Ki = 0.17 nM T88547 C6D5UW 18790190 Ki = 0.38 nM T88547 CBY3Q2 18790194 Ki = 0.28 nM T88547 CWY32U 18790196 Ki = 0.19 nM T88547 CFYK37 18790204 Ki = 4.1 nM T88547 CXA1F2 18790208 Ki = 0.81 nM T88547 C04TCD 18790215 Ki = 190 nM T88547 C53XYC 18790234 Ki = 0.26 nM T88547 CCU7M5 18790248 Ki = 2.3 nM T88547 C2A7IW 18790250 Ki = 6.8 nM T88547 C71TDI 18790258 Ki = 0.29 nM T88547 CT8Y7L 18790272 Ki = 0.32 nM T88547 CF50XE 18790283 Ki = 1.5 nM T88547 C8W2PU 18959700 IC50 = 210 nM T88547 CZY57S 18959702 IC50 = 54 nM T88547 CX3BD8 18959714 IC50 = 58 nM T88547 CZFE27 18959715 IC50 = 118 nM T88547 C7Y2PB 18959716 IC50 = 263 nM T88547 C7Q1KM 18959727 IC50 = 91 nM T88547 C60MOL 18959733 IC50 = 195 nM T88547 CKUS01 18959739 IC50 = 54 nM T88547 CW8PK0 19022852 Ki = 5 nM T88547 COZ07Y 19093638 IC50 = 7.586 nM T88547 CS7A4F 19427051 IC50 = 72 nM T88547 C9KH6O 19427053 IC50 = 9 nM T88547 C4MGT6 19427060 IC50 = 6 nM T88547 C4T9LZ 19606389 IC50 = 210 nM T88547 C1YXZ6 20068647 IC50 > 49 nM T88547 CLH0Z3 20068655 IC50 = 89 nM T88547 C40JIT 21474204 Ki = 5 nM T88547 CRT1Q8 21481466 Ki = 17 nM T88547 C3T5HF 21509921 Ki = 6143 nM T88547 CT7XG9 21830793 Ki = 59 nM T88547 CD5ZM4 21846520 Ki = 74 nM T88547 C2PEQ0 21968329 Ki = 45 nM T88547 CYM17I 22024852 Ki = 9.6 nM T88547 C1I4MZ 22413499 Ki = 2 nM T88547 CVGW27 22875688 Ki = 1.08 nM T88547 CIL6K7 22875693 Ki = 2.53 nM T88547 C72YBR 22875695 Ki = 1.2 nM T88547 C6E2DA 23465639 Ki = 0.06607 nM T88547 CYE83W 24739748 Ki = 233 nM T88547 CP9LR1 24739752 Ki = 128 nM T88547 CDN32O 24743568 Ki = 39 nM T88547 C6B2QL 24743571 Ki = 80.8 nM T88547 C54VFU 24743572 Ki = 9.5 nM T88547 CC52AB 24743739 Ki = 7.2 nM T88547 C5WGF4 24744816 Ki > 1000 nM T88547 C1SDO5 24744977 Ki = 23.1 nM T88547 CC36WF 24835442 Ki = 9 nM T88547 CDC91N 24839550 Ki = 100 nM T88547 CBGO31 24867245 Ki = 1.8 nM T88547 CET2U8 25005670 IC50 = 3.2 nM T88547 CDZ67U 25006418 IC50 = 48.1 nM T88547 C1OJ8G 25006786 IC50 = 2.9 nM T88547 CWT7P6 25059251 Ki = 2.9 nM T88547 CD7SE4 25060019 Ki = 24 nM T88547 CA1EJ2 25120700 Ki = 392 nM T88547 C1SH4X 25167085 Ki = 4.5 nM T88547 CX7QS0 25167087 Ki = 2.1 nM T88547 C90IWB 25184808 Ki = 5484 nM T88547 CWQ5S7 27148262 Ki = 4.3 nM T88547 C4MRQ0 27842480 Ki = 383 nM T88547 CUVS17 29048070 Ki = 2.9 nM T88547 CNK45Q 29150590 Ki = 41 nM T88547 C85BLI 30675158 Ki = 21 nM T88547 CR9N7G 30853613 Ki = 23 nM T88547 C7EJK2 31588412 Ki = 1.9 nM T88547 CO9HV7 40624141 Ki = 42 nM T88547 CRJ5E1 41306333 Ki = 47 nM T88547 CCF93H 41306385 Ki = 3.9 nM T88547 CQSO71 41306434 Ki = 24 nM T88547 CGO25K 41306445 Ki = 10 nM T88547 C83TBP 41307231 Ki = 2.9 nM T88547 CNY78F 42601649 IC50 = 954.99 nM T88547 CJH9I7 42601650 IC50 = 12.88 nM T88547 C7X6FE 42601651 IC50 = 4.467 nM T88547 CFB67A 42601652 IC50 = 58.88 nM T88547 C5J4MX 42601814 IC50 = 5.495 nM T88547 C8WNV1 42601815 IC50 = 17.38 nM T88547 CD81XZ 43267406 IC50 > 100000 nM T88547 CYI6L0 44248689 Ki > 100 nM T88547 CT1R7P 44270247 Ki = 100 nM T88547 C71EWU 44270248 Ki = 2000 nM T88547 C1CMA5 44272667 Ki = 17.7 nM T88547 C7ZMY2 44272754 Ki = 5.7 nM T88547 C5X7RV 44272941 Ki = 30 nM T88547 CBV83R 44272942 Ki = 0.9 nM T88547 C12IYN 44273058 Ki = 5.8 nM T88547 C8CEB5 44273063 Ki = 0.48 nM T88547 CU1HB5 44273339 Ki = 135 nM T88547 C6UN9B 44273356 Ki = 8.6 nM T88547 CQ35UT 44273357 Ki = 19.4 nM T88547 CU71HE 44273383 Ki = 130 nM T88547 C1M4OC 44273461 Ki = 124 nM T88547 CBH0I3 44285300 IC50 = 928 nM T88547 C1MV9C 44285320 IC50 = 63 nM T88547 CVP97C 44285332 IC50 = 65 nM T88547 C4DZY7 44285419 IC50 = 130 nM T88547 CCD68A 44285462 IC50 = 16 nM T88547 CQ4U7F 44285482 Ki = 31.8 nM T88547 CK70ZR 44285702 IC50 = 1630 nM T88547 CWJ9C4 44285740 IC50 = 99 nM T88547 CTR39Y 44291865 Ki = 34 nM T88547 CG1AV3 44292277 Ki = 270 nM T88547 CRT6Q8 44292278 Ki = 300 nM T88547 CVHM52 44292312 Ki = 120 nM T88547 C6PZU2 44292354 Ki = 1 nM T88547 C4H6US 44296111 Ki = 115 nM T88547 CGM01C 44296419 Ki = 456 nM T88547 CT4OF7 44296433 Ki = 161 nM T88547 C6QL4P 44296593 Ki = 49 nM T88547 CM92GY 44296633 Ki = 245 nM T88547 CL5CV9 44296635 Ki = 49 nM T88547 CBGJ28 44296645 Ki > 3300 nM T88547 C7ICW0 44296647 Ki = 241 nM T88547 CWZ4L2 44296655 Ki = 14 nM T88547 C0CS2T 44296665 Ki > 3300 nM T88547 C9GE4U 44297117 Ki > 1000 nM T88547 CMY2U8 44298009 Ki = 8.3 nM T88547 CZL87E 44303090 Ki = 1.7 nM T88547 CTBP60 44303758 Ki = 28 nM T88547 CN5B1M 44304225 IC50 = 4.677 nM T88547 CZA85U 44304236 IC50 = 6.607 nM T88547 CPV5R8 44304238 IC50 = 7.079 nM T88547 CRQ62S 44304240 IC50 = 16.6 nM T88547 CZ9IE3 44304242 IC50 = 81.28 nM T88547 C5DZ7S 44304251 IC50 = 0.2512 nM T88547 C04AXY 44304253 IC50 = 1.175 nM T88547 CWK5I3 44304261 IC50 = 4.571 nM T88547 CRK8S1 44304359 IC50 = 1.738 nM T88547 CIMW61 44304370 IC50 = 2.042 nM T88547 CY9L8D 44304372 IC50 = 2.455 nM T88547 C97XJP 44304406 IC50 = 8.71 nM T88547 C83NIJ 44304409 IC50 = 97.72 nM T88547 C90SZX 44304411 IC50 = 1.995 nM T88547 CNW1J7 44304414 IC50 = 1.82 nM T88547 CF96TW 44304421 IC50 = 2.291 nM T88547 CH2IG4 44304429 IC50 = 2.188 nM T88547 CNS9U4 44304433 IC50 = 4.266 nM T88547 C64ZWJ 44304443 IC50 = 3.467 nM T88547 CEJ6O9 44304447 IC50 = 0.3236 nM T88547 C4BHF5 44304618 IC50 = 2.57 nM T88547 C8Z3WP 44307427 IC50 = 9 nM T88547 CGZ1J8 44307523 Ki = 1.78 nM T88547 C7PZH9 44309297 Ki = 19 nM T88547 COHQ97 44309298 Ki = 8.4 nM T88547 CB2HT7 44309448 Ki = 1140 nM T88547 CT1E5L 44309453 Ki = 6220 nM T88547 C9Y7AI 44309455 Ki = 4 nM T88547 C7HA6I 44309464 Ki = 695 nM T88547 CJN2V0 44309466 Ki = 26 nM T88547 C38TNP 44309468 Ki = 324 nM T88547 C74QMW 44309492 Ki = 4150 nM T88547 C70WAV 44309628 Ki = 5130 nM T88547 CGYQ08 44309667 Ki = 11 nM T88547 C1Q4JD 44309690 Ki = 462 nM T88547 C1MH5F 44309692 Ki = 35 nM T88547 CL3F0P 44309694 Ki = 30 nM T88547 CA98DZ 44309696 Ki = 24 nM T88547 C0QFX9 44309716 Ki = 12 nM T88547 CD8RJ0 44309721 Ki = 0.59 nM T88547 CDB5R0 44309737 Ki = 49 nM T88547 C3YF2M 44309781 Ki = 3 nM T88547 CX5DU2 44309807 Ki = 232 nM T88547 CN0CZ1 44309809 Ki = 4000 nM T88547 CMJ95H 44309824 Ki = 580 nM T88547 CV65SY 44309831 Ki = 17 nM T88547 CX8H4A 44309835 Ki = 384 nM T88547 CT8L0X 44309837 Ki = 32 nM T88547 CG97RP 44309852 Ki = 4520 nM T88547 CT37BP 44309854 Ki = 3500 nM T88547 CE2QW0 44309866 Ki = 8110 nM T88547 C51RVN 44309974 Ki = 223 nM T88547 CCQN61 44309978 Ki = 6 nM T88547 C4UZG0 44309993 Ki = 1 nM T88547 CLYS40 44309995 Ki = 1 nM T88547 CH86ST 44310013 Ki = 298 nM T88547 C9LHD4 44310018 Ki = 214 nM T88547 CUC5I7 44310027 Ki = 16 nM T88547 C03FIO 44310034 Ki = 44 nM T88547 CU0EA9 44310036 Ki = 16 nM T88547 CJYR45 44310038 Ki = 9 nM T88547 C7M5HP 44310050 Ki = 4 nM T88547 C09JTN 44310052 Ki = 4 nM T88547 C4MD0R 44310071 Ki = 2 nM T88547 CY6O4H 44310073 Ki = 1 nM T88547 CN19YU 44310110 Ki = 7500 nM T88547 CL8D2O 44310124 Ki = 90 nM T88547 C4FS9Q 44310126 Ki = 163 nM T88547 CKVO42 44310128 Ki = 20000 nM T88547 CI2TN6 44310145 Ki = 4 nM T88547 COQW09 44310585 Ki = 0.13 nM T88547 C6FM0E 44310664 Ki = 0.8 nM T88547 CRK70Y 44310683 Ki = 1.1 nM T88547 C56NHS 44310857 Ki = 0.66 nM T88547 CWX0S8 44310858 Ki = 0.48 nM T88547 C2VTJ3 44310861 Ki = 0.89 nM T88547 CN08YO 44310878 Ki = 1.3 nM T88547 C6L2KD 44310879 Ki = 1.4 nM T88547 CBVZ21 44310961 Ki = 1.9 nM T88547 C42QYO 44311177 Ki = 7300 nM T88547 C6BX5O 44311179 Ki = 30 nM T88547 C6HEB9 44311180 Ki = 7500 nM T88547 C02DAJ 44311195 Ki = 4 nM T88547 CH7Q9A 44311197 Ki = 5 nM T88547 CBZ06X 44311211 Ki = 1 nM T88547 C5YNX7 44311359 Ki = 1830 nM T88547 C6D5TP 44311361 Ki = 1590 nM T88547 C7VW2Z 44311445 Ki = 6880 nM T88547 C71HBP 44311480 Ki = 6 nM T88547 CRW2P1 44311482 Ki = 7 nM T88547 CCNT08 44311493 Ki = 352 nM T88547 CW8S4Z 44311613 Ki = 4 nM T88547 CO2P4D 44311615 Ki = 70 nM T88547 C3QI6S 44311621 Ki = 10 nM T88547 C9GN7W 44311623 Ki = 13 nM T88547 CTR73J 44311625 Ki = 34 nM T88547 C5IKM9 44311640 Ki = 131 nM T88547 CKMJ50 44312948 Ki = 64 nM T88547 C74HMA 44313623 Ki = 1.33 nM T88547 C3J7XK 44313729 Ki = 1.67 nM T88547 CP3IG8 44313766 Ki = 3 nM T88547 CUQ94M 44313811 Ki = 2.87 nM T88547 C6CTR9 44313813 Ki = 2.87 nM T88547 CYI1A5 44313950 Ki = 0.55 nM T88547 C09MRS 44314013 Ki = 9.04 nM T88547 C4YT2K 44314123 Ki = 1.7 nM T88547 CSX31U 44314127 Ki = 174 nM T88547 CR24KE 44314136 Ki = 1.6 nM T88547 CR2YW9 44314137 Ki = 78 nM T88547 CW79CE 44314138 Ki = 16.3 nM T88547 C8T6GO 44314139 Ki = 154 nM T88547 CIYN38 44314217 Ki = 80 nM T88547 C5DS0N 44314218 Ki = 607 nM T88547 CU27RC 44314387 Ki = 119 nM T88547 CH4R7E 44314603 Ki = 1.7 nM T88547 CJL61P 44315181 Ki = 90 nM T88547 CLCN19 44315510 Ki = 1 nM T88547 CC57FY 44315535 Ki = 5 nM T88547 CEU56A 44315536 Ki = 8 nM T88547 C2DB7M 44315537 Ki = 18 nM T88547 C06BLA 44315552 Ki = 4 nM T88547 CI9GC2 44315578 Ki = 212 nM T88547 CW2I9R 44315579 Ki = 28 nM T88547 CF3M9C 44315580 Ki = 12 nM T88547 CSF86X 44315581 Ki = 2 nM T88547 CJ78AN 44315794 Ki = 4 nM T88547 C6B4CM 44315795 Ki = 22 nM T88547 C2WNL8 44315815 Ki = 8 nM T88547 CMRY42 44315830 Ki = 18 nM T88547 CD5R0G 44318068 IC50 = 163 nM T88547 C9UI8D 44318072 IC50 = 120 nM T88547 CT8WG0 44319215 IC50 = 5312 nM T88547 C0IU3Z 44321002 Ki = 104 nM T88547 C7QE2P 44321166 Ki = 97.2 nM T88547 C0M8TC 44321369 Ki = 138 nM T88547 C45HNC 44321397 Ki = 124 nM T88547 C1M7CY 44321499 Ki = 4420 nM T88547 CD8W0B 44321533 Ki = 552 nM T88547 C1E7MU 44321569 Ki = 5720 nM T88547 CEC92Q 44321621 Ki = 11.1 nM T88547 CAUB15 44321622 Ki = 32.5 nM T88547 CQ5V8G 44321623 Ki = 29.6 nM T88547 C2IAK4 44321648 Ki = 596 nM T88547 CT7X9G 44327682 Ki = 5.86 nM T88547 C61RYB 44327700 Ki = 0.45 nM T88547 CP0OM3 44327701 Ki = 1.04 nM T88547 CLY6O9 44327702 Ki = 3.07 nM T88547 CR9K2G 44327733 Ki = 1.75 nM T88547 C7ECV6 44330983 Ki = 157 nM T88547 CA9YX4 44330991 Ki = 158.49 nM T88547 CNB74Y 44332157 Ki = 35.2 nM T88547 CG4HV0 44332382 Ki = 2.62 nM T88547 CT0C6R 44332389 Ki = 37.4 nM T88547 C52MIY 44332475 Ki = 70.6 nM T88547 C3QS4R 44332496 Ki = 120 nM T88547 CE9JG2 44332500 Ki = 231 nM T88547 CGF56B 44332508 Ki = 1.72 nM T88547 CG2BJ0 44332511 Ki = 71.5 nM T88547 C8L0CI 44332512 Ki = 68.6 nM T88547 CRW57S 44332515 Ki = 1.75 nM T88547 CIZ63N 44332579 Ki = 2.49 nM T88547 C3YHZ7 44334079 Ki = 64.9 nM T88547 C13AJE 44334211 Ki = 1.24 nM T88547 C26IAM 44336365 Ki = 21 nM T88547 CWQ04R 44336430 Ki = 300 nM T88547 C24UOF 44336449 Ki = 2090 nM T88547 C1UWR7 44337609 Ki = 5400 nM T88547 C26ITO 44340881 Ki = 2.6 nM T88547 CF94RB 44340893 Ki = 7 nM T88547 C6HED7 44340900 Ki = 5 nM T88547 CQ2M3C 44340915 Ki = 6 nM T88547 CXKI34 44340919 Ki = 4 nM T88547 CUW0O9 44340942 Ki = 8 nM T88547 CWZ0D7 44340945 Ki = 22 nM T88547 CP9J2Y 44341034 Ki = 1500 nM T88547 C1L8EB 44341173 Ki = 58 nM T88547 CK46JF 44341181 Ki = 5 nM T88547 CV62EA 44341349 Ki = 1.1 nM T88547 C4N6GE 44342597 Ki = 32 nM T88547 C0Z9DY 44342598 Ki = 35 nM T88547 CSZ34A 44342661 Ki = 49 nM T88547 CJVN97 44342684 Ki = 12 nM T88547 CP97HW 44342724 Ki = 1.9 nM T88547 C2EQZ1 44342741 Ki = 0.29 nM T88547 CYTQ61 44342743 Ki = 2.3 nM T88547 C0IJN7 44342746 Ki = 2.8 nM T88547 CQ5B8R 44342747 Ki = 38 nM T88547 CW5RB3 44342753 Ki = 1090 nM T88547 C1LQR9 44342754 Ki = 1330 nM T88547 CD3F2N 44342792 Ki = 6 nM T88547 CC1X5F 44342793 Ki = 43 nM T88547 C46PTB 44342843 Ki = 69 nM T88547 CNO76C 44342910 Ki = 18100 nM T88547 C5NQP9 44342911 Ki = 739 nM T88547 CNG79I 44342912 Ki = 45 nM T88547 CLC0Z1 44342925 Ki = 40 nM T88547 C74GDW 44342933 Ki = 104 nM T88547 CG1X6K 44342934 Ki = 16600 nM T88547 C2BPW6 44344745 IC50 = 182 nM T88547 CZV21Q 44347713 Ki = 26 nM T88547 CLG65Q 44347771 Ki = 5 nM T88547 CUI12W 44347787 Ki = 13 nM T88547 C7Q4IB 44347788 Ki = 174 nM T88547 CYP17T 44350537 Ki = 17.49 nM T88547 CD38RO 44350538 Ki = 117 nM T88547 C0K5CR 44350649 Ki = 95.69 nM T88547 CCU89V 44350664 Ki = 34.1 nM T88547 C3CM2E 44350704 Ki = 280.75 nM T88547 C03YVC 44350708 Ki = 249.3 nM T88547 CC3Y4A 44350710 Ki = 302.4 nM T88547 C8EF0H 44350786 Ki = 40.4 nM T88547 C5E3FK 44350787 Ki = 517.7 nM T88547 C41UID 44350800 Ki = 194.5 nM T88547 CRC5I3 44350810 Ki = 240.3 nM T88547 C69MTC 44350812 Ki = 191 nM T88547 CMRX47 44350817 Ki = 175 nM T88547 CZMW86 44350827 Ki = 30.89 nM T88547 CI7KH4 44350870 Ki = 380 nM T88547 C7NC0V 44350885 Ki = 106.8 nM T88547 C60IJH 44350886 Ki = 8.5 nM T88547 C4QP5U 44350942 Ki = 183 nM T88547 C50HVX 44350991 Ki = 32.5 nM T88547 C7FCG1 44351070 IC50 = 1250 nM T88547 C09PFU 44356418 IC50 = 3378 nM T88547 CMP3T6 44356420 IC50 = 130 nM T88547 CL0MH9 44356422 IC50 = 113 nM T88547 CR16SL 44356442 IC50 = 480 nM T88547 CNDC89 44356481 IC50 = 180 nM T88547 C3SZV2 44356483 IC50 = 178 nM T88547 C2GZ4I 44356488 IC50 = 224 nM T88547 CH53UR 44356504 IC50 = 494 nM T88547 C4U6DG 44356510 IC50 = 110 nM T88547 CD0G2I 44356520 IC50 = 112 nM T88547 C1E3PF 44356530 IC50 = 18.2 nM T88547 CBV4R6 44356532 IC50 = 113 nM T88547 CB0G7Y 44356538 IC50 = 221 nM T88547 CEZQ08 44356560 IC50 = 200 nM T88547 C4HJ1Q 44356562 IC50 = 40.2 nM T88547 CR3BG4 44356573 IC50 = 309 nM T88547 C9YHF4 44356579 IC50 = 4.5 nM T88547 C8NM9A 44356581 IC50 = 7.4 nM T88547 CL3EM6 44356583 IC50 = 5.7 nM T88547 CH0Z5S 44356587 IC50 = 45.3 nM T88547 CFUS27 44356589 IC50 = 205 nM T88547 C5W4TO 44356593 IC50 = 30.7 nM T88547 CU0M1F 44356607 IC50 = 15.8 nM T88547 C0IY2M 44356642 IC50 = 8 nM T88547 C5AM0K 44356750 IC50 = 203 nM T88547 CMQV74 44356752 IC50 = 261 nM T88547 CS4HR6 44356757 IC50 = 113 nM T88547 CL9H7O 44356759 IC50 = 1947 nM T88547 CYGJ56 44356761 IC50 = 79 nM T88547 CHRM80 44356783 IC50 = 115 nM T88547 CP1JG7 44356785 IC50 = 755 nM T88547 CE76RV 44356787 IC50 = 421 nM T88547 C8LI5Y 44356836 IC50 = 19.6 nM T88547 C8T9NZ 44356838 IC50 = 17.3 nM T88547 CVY7W0 44356840 IC50 = 23.9 nM T88547 CI2A0J 44357414 IC50 = 949 nM T88547 C35PQS 44357415 IC50 = 1830 nM T88547 CC7V3Q 44361163 Ki = 11.7 nM T88547 CT52YL 44361164 Ki = 31.7 nM T88547 C0XLF9 44361167 Ki = 14.8 nM T88547 CUB80P 44361281 Ki = 3.36 nM T88547 CY3F5S 44361297 Ki = 18.4 nM T88547 C4IZ6C 44361388 Ki = 5.74 nM T88547 CQOD63 44361659 IC50 = 8.5 nM T88547 C97MEH 44362252 Ki = 1.62 nM T88547 CE3KC6 44362800 Ki = 1.71 nM T88547 CHJI46 44364124 Ki = 3600 nM T88547 C6RHC8 44364145 Ki > 10000 nM T88547 CH93PJ 44364189 Ki = 1465 nM T88547 CEG3S1 44364199 Ki = 11.8 nM T88547 CRP3B1 44370359 Ki = 34.5 nM T88547 CF8TC4 44370527 Ki = 109 nM T88547 CCH1J0 44370541 Ki = 58.2 nM T88547 CYF19D 44378807 Ki = 18.6 nM T88547 C14WCF 44385319 IC50 = 9.7 nM T88547 CEY85C 44386517 Ki = 0.7 nM T88547 CX7W3K 44398003 Ki = 74 nM T88547 C2MZH9 44398036 Ki = 0.5 nM T88547 C7C2TW 44398114 Ki = 1 nM T88547 C17XVW 44398137 Ki > 100000 nM T88547 CM45OW 44398162 Ki = 5 nM T88547 C7E9FT 44403183 IC50 = 6.6 nM T88547 C08XKE 44403246 IC50 = 54 nM T88547 CI4J5V 44403247 IC50 = 77 nM T88547 CF6X3K 44460274 IC50 = 250 nM T88547 CZS51T 44460446 IC50 > 10000 nM T88547 CW0J1K 44573133 Ki = 2240 nM T88547 CC6GX9 44573260 Ki = 53 nM T88547 CWAX45 44573261 Ki = 1600 nM T88547 CU4X2D 44818602 Ki = 7.1 nM T88547 C4LOY2 45115589 Ki < 1000 nM T88547 CK5Z6Q 45160790 Ki = 1584.89 nM T88547 C69RIC 45260531 IC50 = 21.38 nM T88547 CEY5U0 45260638 Ki = 2.51 nM T88547 C4I6VA 45262124 IC50 = 82 nM T88547 CDB08V 45262186 IC50 = 30.1 nM T88547 CEYM15 45264502 IC50 = 16.6 nM T88547 C5H0TZ 45487178 Ki = 0.4365 nM T88547 C08PKX 45487184 Ki = 0.08913 nM T88547 CR46EI 45487199 Ki = 0.09772 nM T88547 C1KX4B 45487204 Ki = 0.05754 nM T88547 C4RCU0 45487212 Ki = 0.05248 nM T88547 CP8EI4 45487215 Ki = 0.1096 nM T88547 CT29RN 45489962 Ki = 3200 nM T88547 CKCN84 46225028 Ki = 2280 nM T88547 C34ZXM 46225029 Ki = 149 nM T88547 C46HRG 46877990 IC50 = 928 nM T88547 CN8QY1 46877991 IC50 = 1247 nM T88547 CFE82I 46877992 IC50 = 3650 nM T88547 CC3T9L 46877993 IC50 = 5303 nM T88547 CNW5M8 46877994 IC50 = 3267 nM T88547 CDYS63 46877995 IC50 = 42 nM T88547 CS1X3U 46877996 IC50 = 2670 nM T88547 C7M0RU 46877997 IC50 = 1335 nM T88547 CGN59L 46877998 IC50 = 200 nM T88547 CK5Z0C 46877999 IC50 = 228 nM T88547 C3JG1D 46878000 IC50 = 110 nM T88547 CJD01C 46878001 IC50 = 76 nM T88547 CRB5L6 46878002 IC50 = 870 nM T88547 CK7N6S 46878005 IC50 = 224 nM T88547 CYM6C0 46878006 IC50 = 1155 nM T88547 C85YUM 46878007 IC50 = 1609 nM T88547 CE72KC 46878008 IC50 = 302 nM T88547 CBG9X7 46878009 Ki = 11 nM T88547 CIN90O 46878010 IC50 = 196 nM T88547 CT1MY8 46878011 IC50 = 5952 nM T88547 CHV7E8 46878012 IC50 = 1385 nM T88547 CG98OY 46878013 IC50 = 211 nM T88547 C4T5FE 46878014 IC50 = 208 nM T88547 C3P1JH 46878015 IC50 = 2374 nM T88547 CWM1O2 46878220 Ki = 8554 nM T88547 CQ0J2T 46906592 Ki > 800 nM T88547 CPBM68 46906593 Ki > 800 nM T88547 CE9Y7S 46907276 Ki > 800 nM T88547 CID6G4 46907277 Ki > 800 nM T88547 C9L3ZI 46911069 Ki = 79.43 nM T88547 C1N4ID 49832807 Ki = 194 nM T88547 CWMU78 49853575 IC50 = 590 nM T88547 CLJK94 49853576 IC50 = 270 nM T88547 CC48YF 49853577 IC50 = 1200 nM T88547 CZ4B0R 49853579 IC50 = 210 nM T88547 C3C9EJ 49853580 IC50 > 100000 nM T88547 CTF02Q 49853581 IC50 = 7600 nM T88547 CN8JR2 49853583 IC50 = 15200 nM T88547 CK3S1W 49853672 IC50 = 11500 nM T88547 C98QPG 49853674 IC50 = 18800 nM T88547 CI4W2P 49853676 IC50 = 16300 nM T88547 CPI6N0 49853777 IC50 > 100000 nM T88547 C94GDK 49853778 IC50 > 100000 nM T88547 C85YTF 49853781 IC50 = 15800 nM T88547 CHV3U8 49853881 IC50 = 430 nM T88547 C7MGD9 49853882 IC50 = 7240 nM T88547 CTBY97 49853883 IC50 = 390 nM T88547 CQP63D 49853884 IC50 = 2250 nM T88547 CY8M9A 49853885 IC50 = 8410 nM T88547 CECY14 49853886 IC50 = 21100 nM T88547 CP6GK8 49853980 IC50 = 180 nM T88547 C0J1OX 49853981 IC50 > 100000 nM T88547 CJ0Q5W 49853983 IC50 = 11800 nM T88547 CHK26Y 49853984 IC50 = 930 nM T88547 CJWH91 49853986 IC50 = 18000 nM T88547 CN0JU9 49853987 IC50 = 500 nM T88547 C5OXM4 49854189 IC50 = 11600 nM T88547 C8DVX6 49855131 IC50 = 3250 nM T88547 CTV1K4 49855133 IC50 = 8830 nM T88547 C2RY0J 50878551 Ki = 302 nM T88547 C1W6TV 50898777 Ki = 398.11 nM T88547 CXMZ73 50898778 Ki > 10000 nM T88547 CU63SQ 50994498 Ki = 0.59 nM T88547 CE4KP1 51050257 Ki > 10000 nM T88547 C3A9OY 51111240 Ki = 20 nM T88547 CPJZ31 52149645 Ki = 5.8 nM T88547 C82HKM 52750322 Ki = 3.7 nM T88547 COCZ63 52912210 IC50 = 43 nM T88547 CMJ62D 53245590 Ki = 410 nM T88547 CMOZ61 53475319 Ki = 531 nM T88547 C4BWN0 53707349 Ki = 660 nM T88547 CWK70Q 54315083 Ki = 1640 nM T88547 CECV98 54581003 IC50 = 1.202 nM T88547 C7L9JS 54583594 Ki = 39 nM T88547 CWY64L 54591111 Ki = 83.4 nM T88547 C2Y7LX 54591112 Ki = 296 nM T88547 C3KO4E 56652775 Ki = 1492 nM T88547 CQ3SG5 56656039 Ki = 10320 nM T88547 CJKO58 56852956 Ki = 346.74 nM T88547 C1TC7Q 56963799 Ki > 10000 nM T88547 CXW2C4 57340967 Ki > 1000 nM T88547 CZU6L2 57345618 Ki = 2.884 nM T88547 CK9G8H 57345619 Ki = 3.6 nM T88547 C4EXS6 57396571 Ki = 51.7 nM T88547 CO3B4P 57399494 Ki = 63 nM T88547 CYN38R 57401819 Ki = 36 nM T88547 CZ2UB5 57705473 Ki = 14.2 nM T88547 C0JMC4 57861965 Ki = 879 nM T88547 C3TNQ5 60346448 Ki = 3.6 nM T88547 C7JG9R 60701380 Ki > 100 nM T88547 CW36YC 66561968 Ki = 10000 nM T88547 C7FMA4 70676458 Ki = 5090 nM T88547 CNL86E 70681422 IC50 = 63.3 nM T88547 C5IN6M 70683538 IC50 = 12.4 nM T88547 CNB3C9 70691984 IC50 > 100 nM T88547 C57VRM 70695522 IC50 = 299 nM T88547 C08PHA 70696149 IC50 = 0.27 nM T88547 CUD40A 70697541 IC50 = 9 nM T88547 CR5KY1 71061607 Ki > 5000 nM T88547 C72XPZ 71061659 Ki > 5000 nM T88547 CD1ET2 71061756 Ki > 5000 nM T88547 C5KM2W 71061887 Ki > 5000 nM T88547 CN7C9S 71222835 Ki = 29 nM T88547 C8QWT7 71222908 Ki = 58 nM T88547 C3HSF6 71222985 Ki = 18 nM T88547 C8SDY4 71222995 Ki = 98 nM T88547 CO3PG8 71223000 Ki = 16 nM T88547 CA6KM2 71223037 Ki = 141 nM T88547 CA8NH6 71223095 Ki = 514 nM T88547 CU64JP 71223100 Ki = 55 nM T88547 CN97QC 71223119 Ki = 399 nM T88547 CTC30W 71223161 Ki = 62 nM T88547 CO47LV 71223168 Ki = 371 nM T88547 CY17ZB 71223185 Ki = 116 nM T88547 CY9S4C 71223204 Ki = 11 nM T88547 CA03HG 71223206 Ki = 192 nM T88547 C7YJT8 71223208 Ki = 9 nM T88547 C89SAL 71223232 Ki = 156 nM T88547 C20GSJ 71223247 Ki = 25 nM T88547 CDP92M 71223250 Ki = 41 nM T88547 CGO4J3 71223252 Ki = 51 nM T88547 CFZ29E 71223262 Ki = 79 nM T88547 CW2D8E 71223267 Ki = 9 nM T88547 CEIG57 71223275 Ki = 32731 nM T88547 CU49ST 71223296 Ki = 23 nM T88547 CO19CM 71223298 Ki = 181 nM T88547 CS39DP 71223393 Ki = 716 nM T88547 CIMT57 71223397 Ki = 33 nM T88547 C8YB9W 71223407 Ki = 818 nM T88547 C02UWQ 71223427 Ki = 292 nM T88547 C3XTM8 71223439 Ki = 24 nM T88547 CLN1Q4 71223454 Ki = 119 nM T88547 CZR75D 71223459 Ki = 21 nM T88547 CY5K3O 71223493 Ki > 1000 nM T88547 C0W4UT 71223519 Ki = 100 nM T88547 C7KZ9O 71225558 Ki = 740 nM T88547 CL3E7G 71225577 Ki = 45 nM T88547 CDG9F6 71225600 Ki = 42923 nM T88547 C90WEH 71225643 Ki = 165 nM T88547 C32CRY 71225858 Ki = 6194 nM T88547 CW6IJ4 71225871 Ki = 200 nM T88547 CUYA72 71225882 Ki = 85 nM T88547 C3A5GS 71225888 Ki = 813 nM T88547 C47ZXI 71225920 Ki = 184 nM T88547 C7R0VL 71225947 Ki = 12 nM T88547 C2ZP6M 71225970 Ki = 946 nM T88547 CP9N6I 71225996 Ki = 294 nM T88547 C8B4HC 71226084 Ki = 13803 nM T88547 C8Y9VF 71226102 Ki = 112 nM T88547 CXG39S 71226177 Ki = 25770 nM T88547 C5MX6Z 71226198 Ki = 18000 nM T88547 CDTW51 71226340 Ki = 108 nM T88547 COY7Z0 71231455 Ki = 55 nM T88547 CCO7J6 71449812 Ki = 99.1 nM T88547 CDP7T0 71449813 Ki = 44 nM T88547 CXO90E 71449814 Ki = 139 nM T88547 CE3SF8 71449822 Ki = 8.9 nM T88547 CYLG97 71451628 Ki = 8.6 nM T88547 C3IN7Y 71451629 Ki = 13.3 nM T88547 CYG43C 71451630 Ki = 9.4 nM T88547 COL29E 71451631 Ki = 8.4 nM T88547 C0OBW8 71451632 Ki = 14.8 nM T88547 C2ENG0 71451633 Ki = 8.5 nM T88547 C4TWS5 71452172 Ki = 4.1 nM T88547 C26HJP 71452705 IC50 = 897 nM T88547 CPU9L0 71453455 Ki > 1000 nM T88547 C29CJD 71453456 Ki = 17.8 nM T88547 CG72SV 71453464 Ki = 16.5 nM T88547 C2IZQ3 71454076 IC50 = 12.3 nM T88547 CW3K2A 71455165 Ki = 65 nM T88547 CZ4HI3 71455166 Ki = 33.8 nM T88547 CMYL95 71455809 IC50 = 36.1 nM T88547 CE5K0Q 71456164 Ki = 762.3 nM T88547 CD0X6R 71456959 Ki > 1000 nM T88547 C4ZW0F 71457595 IC50 = 5.2 nM T88547 C1YGK5 71459491 IC50 = 2.9 nM T88547 CF8TR1 71459493 IC50 = 42 nM T88547 COE9Z8 71460635 Ki = 180 nM T88547 CZH53R 71460636 Ki = 33.3 nM T88547 C96HIW 71460640 Ki = 16.1 nM T88547 C2W9ZQ 71462356 Ki = 18.9 nM T88547 CK40DZ 71462357 Ki = 9.6 nM T88547 C0KR7M 71487770 Ki = 9 nM T88547 C63XQF 71487772 Ki = 22 nM T88547 CGB8N6 71488612 Ki = 13 nM T88547 C91OQB 71503148 Ki = 7 nM T88547 CK54BX 71601215 Ki = 1250 nM T88547 CBO95T 71601216 Ki = 1700000 nM T88547 C2S4EK 71654693 Ki = 536 nM T88547 CJ1S3B 71654694 Ki = 317 nM T88547 CGB32Z 71654695 Ki = 15 nM T88547 C6ZV8T 71655284 Ki = 194 nM T88547 CRFG67 71655285 Ki > 1000 nM T88547 CPOU74 71655286 Ki = 377 nM T88547 C29WRX 71655287 Ki > 1000 nM T88547 CQ70ER 71655288 Ki > 1000 nM T88547 CPW26Z 71655347 Ki = 79 nM T88547 CT8J6R 71655349 Ki > 1000 nM T88547 C0M8WK 71655351 Ki > 1000 nM T88547 CS31VA 71655413 Ki = 19 nM T88547 C0JQL7 71655415 Ki > 1000 nM T88547 CELM32 71655416 Ki = 178 nM T88547 CX72JE 71655418 Ki = 14 nM T88547 C8YHC4 71655477 Ki > 1000 nM T88547 CUHP20 71655478 Ki > 1000 nM T88547 CCD58E 71655480 Ki > 1000 nM T88547 CQIT18 71655541 Ki > 1000 nM T88547 CZN13Q 71655543 Ki > 1000 nM T88547 C94IXE 71655545 Ki > 1000 nM T88547 C7GP2C 71655610 Ki = 302 nM T88547 CL89HF 71655612 Ki = 245 nM T88547 CD78YO 71655614 Ki > 1000 nM T88547 CF78EW 71655616 Ki = 108 nM T88547 C9JF3X 71655681 Ki = 410 nM T88547 CVL20F 71655683 Ki = 67 nM T88547 CF9G8Q 71655685 Ki > 1000 nM T88547 CJ14RU 71655744 Ki > 1000 nM T88547 C6XU2K 71655746 Ki = 124 nM T88547 CDL35U 71655748 Ki = 30 nM T88547 CD63JO 71716506 Ki > 1000 nM T88547 C9M1OY 71716507 Ki = 6.3 nM T88547 CI3OB7 71717119 Ki = 2.75 nM T88547 CWOC31 71718342 Ki > 1000 nM T88547 CDN18F 72950534 Ki = 46.08 nM T88547 C8R1CQ 72950535 Ki = 13.36 nM T88547 C62XVD 72950697 Ki = 45.32 nM T88547 CJZW17 72950698 Ki = 38 nM T88547 CBV3X0 72950699 Ki > 1000 nM T88547 CX93FC 73056461 Ki = 34 nM T88547 CGDH92 73056753 Ki = 29 nM T88547 CC65OA 73213195 Ki > 10000 nM T88547 CW83DK 73213196 Ki = 218.78 nM T88547 CO79PJ 73345319 Ki = 40 nM T88547 CCV91B 73346042 Ki > 10000 nM T88547 C36ZPL 73350500 IC50 = 15200 nM T88547 C5X6WV 73353481 IC50 = 86800 nM T88547 CNA59Q 73354414 Ki = 38.9 nM T88547 C6P0HF 74766963 Ki = 100 nM T88547 CWK67L 74766964 Ki = 74 nM T88547 CWI54G 74766966 Ki = 82 nM T88547 C43THL 74766967 Ki = 732 nM T88547 C42MEP 74767042 Ki = 72 nM T88547 C9F2RU 74767046 Ki = 707 nM T88547 C1S8MT 74767047 Ki = 40.74 nM T88547 C6EX3U 74767048 Ki = 112 nM T88547 CAE45U 74767050 Ki = 666 nM T88547 CK3B4H 74767125 Ki = 300 nM T88547 CS2R9T 74767126 Ki = 95 nM T88547 CJ1W9E 74767127 Ki = 531 nM T88547 CPD9C5 74767128 Ki = 137 nM T88547 CV6KE8 74767129 Ki = 558 nM T88547 C7YR5T 74767130 Ki = 447 nM T88547 CI1GQ0 74767131 Ki = 926 nM T88547 CXLO16 74767207 Ki = 35 nM T88547 CK7WU2 74767208 Ki = 43 nM T88547 C98KAZ 74767209 Ki = 709 nM T88547 CE7RM5 74767211 Ki = 802 nM T88547 CX13JM 74767212 Ki = 31 nM T88547 C94IPS 74767213 Ki = 63 nM T88547 CAY81N 74767285 Ki = 31 nM T88547 C2SR1H 74767286 Ki = 39 nM T88547 C3FVE7 74767287 Ki = 48 nM T88547 C8RV5C 74767288 Ki = 11843 nM T88547 CVLI72 74767289 Ki = 9460 nM T88547 C7CIB1 74767290 Ki = 23832 nM T88547 CDA4B3 74767291 Ki = 1834 nM T88547 C0VXI7 74767363 Ki = 76 nM T88547 C4DEJ0 74767364 Ki = 475 nM T88547 CP92AE 74767365 Ki = 2915 nM T88547 CI61EO 74767366 Ki = 125 nM T88547 CY3AM9 74767367 Ki = 93 nM T88547 CK14JY 74767368 Ki = 1717 nM T88547 C8HA0F 74767448 Ki = 715 nM T88547 C2E7QW 75201901 Ki = 8200 nM T88547 CQ71AT 76073628 Ki = 5 nM T88547 C3AD4C 76313525 Ki = 0.91 nM T88547 C28RIZ 76518514 Ki = 21.88 nM T88547 CQ3EY1 76683576 Ki = 818 nM T88547 C5PW6K 76683678 Ki = 49 nM T88547 CXM51U 76683680 Ki = 31 nM T88547 CGE15Z 76683773 Ki = 46 nM T88547 CL03DO 76683775 Ki = 97 nM T88547 C8HAR3 76683777 Ki = 61 nM T88547 C1EY3H 76683779 Ki > 1000 nM T88547 CG0TR9 76683781 Ki = 10 nM T88547 C3O2FD 76683785 Ki = 781 nM T88547 C95OWP 76683875 Ki = 9 nM T88547 C01RIY 76683877 Ki = 12 nM T88547 C7SN9G 76683881 Ki = 9616 nM T88547 C67SLP 76683883 Ki = 23 nM T88547 C6IS1X 76683885 Ki = 52 nM T88547 CBSD29 76683976 Ki = 35 nM T88547 C1W4ER 76683978 Ki = 701 nM T88547 CITA80 76683982 Ki = 194 nM T88547 CC5J3B 76683988 Ki = 56 nM T88547 C0WR4O 76684092 Ki = 36 nM T88547 CJ1KN0 76684094 Ki = 13 nM T88547 C2XSM8 76684096 Ki = 878 nM T88547 CR76SA 76684100 Ki = 33 nM T88547 CLD49W 76684104 Ki = 62 nM T88547 C08EZV 76684202 Ki = 46 nM T88547 CGBP93 76684204 Ki > 1000 nM T88547 C75VCS 76684206 Ki = 70 nM T88547 CKC14S 76684208 Ki = 105 nM T88547 CV62NT 76684214 Ki = 58 nM T88547 CXO78M 76684294 Ki = 144 nM T88547 C8P7EC 76684296 Ki = 31 nM T88547 CG6C3U 76684304 Ki = 275 nM T88547 C1EF6U 76684306 Ki = 459 nM T88547 CB95UF 76684383 Ki = 388 nM T88547 C6MSH2 76684391 Ki = 111 nM T88547 C5VNK9 76684473 Ki > 1000 nM T88547 C2EO6P 76684475 Ki = 451 nM T88547 CI21ES 76684477 Ki = 216 nM T88547 COY67V 76684479 Ki = 241 nM T88547 CC81FG 76684481 Ki = 273 nM T88547 CI6K1G 76684564 Ki = 508 nM T88547 CLR0B8 78043801 Ki = 15 nM T88547 CZ75NQ 86582973 Ki = 51 nM T88547 CC0IB7 90146004 Ki = 112 nM T88547 CKH16N 90146246 Ki = 634 nM T88547 CY14OV 90269112 Ki = 662 nM T88547 C68URF 90269115 Ki > 1000 nM T88547 CM90FD 90643603 Ki = 7463 nM T88547 C5B8PY 90643604 Ki = 3063 nM T88547 CPN65E 90643787 IC50 = 30000 nM T88547 CLM0J5 90644067 Ki = 1148 nM T88547 CG83SL 90654976 Ki = 10 nM T88547 C4UEJ8 90654977 Ki = 3063 nM T88547 C5O4JQ 90654978 Ki = 10.5 nM T88547 C5IE8A 90655529 Ki = 29 nM T88547 C2SMQ1 90655530 Ki = 7.5 nM T88547 C7QRC3 90655531 Ki = 6.8 nM T88547 CK8M5I 90655532 Ki = 27 nM T88547 CZVJ18 90655533 Ki = 279 nM T88547 C1PAN6 90655534 Ki = 107 nM T88547 CU8FY3 90655535 Ki = 711 nM T88547 C6KXQ7 90655536 Ki = 465 nM T88547 CI35AY 90655537 Ki = 491 nM T88547 C8TOW0 90666080 Ki = 158.49 nM T88547 C2HF4P 90666081 Ki = 125.89 nM T88547 C1E9BD 90666082 Ki = 63.1 nM T88547 CH4Q1J 90666083 Ki = 63.1 nM T88547 COS08L 90666084 Ki = 1258.93 nM T88547 C1WUZ3 90666085 Ki = 398.11 nM T88547 CYUV14 90666086 Ki = 15.85 nM T88547 C9SMH8 90666087 Ki = 10 nM T88547 CZPD45 90666088 Ki = 25.12 nM T88547 CZX94Q 90666089 Ki = 630.96 nM T88547 C34WZM 90666090 Ki = 25.12 nM T88547 CT21RI 90666091 Ki = 199.53 nM T88547 CIBZ73 90666092 Ki = 100 nM T88547 CO7I5L 90666093 Ki = 79.43 nM T88547 CH5R8Q 98049507 Ki = 6300 nM T88547 C2EJK6 101910737 Ki = 1.1 nM T88547 CB5DK1 102004349 Ki = 6 nM T88547 CO6Z7J 110440208 Ki = 1.6 nM T88547 CBW0U9 110445832 Ki = 1.4 nM T88547 C5CDE0 118562359 Ki = 28 nM T88547 CS63OE 118562362 Ki = 209 nM T88547 CWH9B5 118562372 Ki = 91 nM T88547 C60BSA 118562375 Ki = 10 nM T88547 CE3D0A 118562384 Ki = 8 nM T88547 C7IVW9 118562402 Ki = 54 nM T88547 C63EGC 118562428 Ki = 53 nM T88547 CE53DJ 118562440 Ki = 8 nM T88547 CW26NV 118562451 Ki = 14 nM T88547 C7G5HO 118562469 Ki = 54 nM T88547 C3BIL8 118562502 Ki = 68 nM T88547 C5JKQ9 118562510 Ki = 6 nM T88547 C12CKV 118562522 Ki = 14 nM T88547 CF6LK7 118562538 Ki = 9 nM T88547 C6FOS9 118562556 Ki = 15 nM T88547 C25MXS 118562567 Ki = 11 nM T88547 C3TQE7 118562573 Ki = 88 nM T88547 CJF1E6 118562576 Ki = 40 nM T88547 C5QB2S 118562584 Ki = 21 nM T88547 C6TC3D 118562598 Ki = 53 nM T88547 CWA4B2 118562606 Ki = 13 nM T88547 C2EPN1 118565438 Ki = 99 nM T88547 C0XIN5 118567313 Ki = 32 nM T88547 C6PA1C 118567531 Ki = 103 nM T88547 CD4XK8 118567534 Ki = 14 nM T88547 CLVO18 118567538 Ki = 63 nM T88547 C1CP6Z 118567543 Ki = 58 nM T88547 C32PGF 118567545 Ki = 48 nM T88547 C7G8IT 118567547 Ki = 3 nM T88547 CN1DU3 118567549 Ki = 275 nM T88547 CKQ15C 118567550 Ki = 122 nM T88547 CJ43GO 118567552 Ki = 55 nM T88547 CV7U9Y 118567593 Ki = 237 nM T88547 CXW0K9 118567604 Ki = 11 nM T88547 C4ULH8 118567605 Ki = 13 nM T88547 C7DO6S 118567606 Ki = 13 nM T88547 C8TP7C 118567608 Ki = 8 nM T88547 C70RDE 118567618 Ki = 51 nM T88547 CGN3Z4 118567654 Ki = 26 nM T88547 CJOK48 118567670 Ki = 57 nM T88547 C4GDV1 118567672 Ki = 112 nM T88547 CK5T2Z 118567678 Ki > 1000 nM T88547 CCY60Z 118567689 Ki = 622 nM T88547 C59GUQ 118567742 Ki = 9 nM T88547 C36JSR 118567743 Ki = 8 nM T88547 C5NI2E 118567744 Ki = 38 nM T88547 CI0JY2 118567747 Ki = 39 nM T88547 CHU07G 118607283 Ki = 1.2 nM T88547 CX2QI6 118607309 Ki = 3.6 nM T88547 CIW02L 118607351 Ki = 4.3 nM T88547 C84QJX 118607364 Ki = 1.1 nM T88547 CX5B2A 118607439 Ki = 6.5 nM T88547 CXOT38 118607453 Ki = 7.3 nM T88547 C4U2GB 118607455 Ki = 1.7 nM T88547 CSB25E 118709750 Ki = 70.79 nM T88547 CD4S9R 118709751 Ki = 57 nM T88547 C4XS8G 118724294 Ki = 5.3 nM T88547 CG6O7M 118724295 Ki = 6.2 nM T88547 CLNB04 118724296 Ki = 4.3 nM T88547 CJ47XE 118724297 Ki = 18 nM T88547 CDL21J 118724298 Ki = 2 nM T88547 CT2RJ5 118724299 Ki > 200 nM T88547 C64SLY 118724300 Ki = 28 nM T88547 CK3RS5 118724301 Ki = 72 nM T88547 CC5E1Q 118724302 Ki = 160 nM T88547 CCE9F4 118724303 Ki = 7.2 nM T88547 CZC13F 118724304 Ki = 11 nM T88547 CQI71Z 118724305 Ki = 11 nM T88547 CJ1VY3 118724306 Ki = 2.5 nM T88547 C9ZR4V 118724307 Ki = 18 nM T88547 CR05GL 118724308 Ki = 11 nM T88547 CT36KB 118724309 Ki > 200 nM T88547 CTU50G 118724310 Ki = 36 nM T88547 CHP0Q2 118724311 Ki = 8 nM T88547 C5W8KO 118724312 Ki = 8.4 nM T88547 C8L5HP 118724313 Ki = 72 nM T88547 CHBZ37 118724314 Ki = 11 nM T88547 CYE4H7 118724315 Ki > 200 nM T88547 C1OHA6 118724316 Ki = 12 nM T88547 CTE58Z 118730369 Ki = 200 nM T88547 C3SL6R 118731566 Ki = 5.3 nM T88547 CSZ3F7 118731567 Ki = 1.2 nM T88547 C1TUD2 118731568 Ki = 0.9 nM T88547 C3NUS9 118731569 Ki = 6.4 nM T88547 C9WKE6 118731570 Ki = 10.3 nM T88547 CSZ4K3 118731571 Ki = 3.1 nM T88547 C1N6GY 118731572 Ki = 0.6 nM T88547 CMC9X4 118731573 Ki = 4.7 nM T88547 CL5H9N 118731574 Ki > 100 nM T88547 CSI32D 118731575 Ki = 2.2 nM T88547 CA8DB0 118731576 Ki > 100 nM T88547 CD01IE 118731577 Ki > 100 nM T88547 C5PXE8 118731578 Ki > 100 nM T88547 CNK9U1 118731579 Ki > 100 nM T88547 C8P6OB 118731580 Ki = 30.3 nM T88547 CT1G4C 118731581 Ki = 5.7 nM T88547 C6Q4SP 118731582 Ki > 100 nM T88547 CWE78H 118731583 Ki > 100 nM T88547 CH3TQ1 118732991 IC50 = 135 nM T88547 C7ODW3 122195524 Ki < 300 nM T88547 C5QIE8 124197459 Ki = 133 nM T88547 C09PAE 126744799 Ki = 205 nM T88547 COJ60B 126744800 Ki = 147 nM T88547 C2U4GO 126744949 Ki = 656 nM T88547 C0FKA4 126744972 Ki = 61 nM T88547 C79BZK 127026013 Ki = 31 nM T88547 C9E4NV 127026014 Ki = 2200 nM T88547 CTBN56 127026052 Ki = 85.11 nM T88547 C64OKQ 127027941 Ki = 676 nM T88547 CJ4YC0 127031397 Ki = 119 nM T88547 CBU9G2 127031398 Ki = 37 nM T88547 CE1IA7 127031399 Ki = 53 nM T88547 C4WKG9 127031403 Ki = 12 nM T88547 CEDM28 127031404 Ki = 130 nM T88547 CV5UH0 127031405 Ki = 350 nM T88547 CHN9X2 127031422 Ki = 124 nM T88547 C0CY9W 127031423 Ki = 57 nM T88547 CNH2V8 127031424 Ki = 13 nM T88547 C2W0HL 127031949 Ki = 122 nM T88547 CU49VE 127036186 Ki = 74.13 nM T88547 CG06BD 127036932 Ki = 97.72 nM T88547 CVW71O 127036953 Ki = 102.33 nM T88547 C9M5RN 127048369 Ki = 73 nM T88547 CLM5O3 127048370 Ki = 27 nM T88547 C6J3FW 127048371 Ki = 24 nM T88547 C1AX7T 127050366 Ki = 6 nM T88547 C8VKE5 127050367 Ki = 27 nM T88547 CH64PD 127050993 Ki = 2.4 nM T88547 C1UPC8 127050994 Ki = 2.8 nM T88547 CVH86Y 127050995 Ki = 1.6 nM T88547 CM3I6O 127051201 Ki = 6.4 nM T88547 C1CA7B 127051216 Ki = 2.2 nM T88547 C6L5ZK 127051267 Ki = 13 nM T88547 CB8W3Y 127051268 Ki = 7.2 nM T88547 CH3SP2 127051269 Ki = 38 nM T88547 CX3KP6 127051889 Ki = 3.2 nM T88547 C50GOC 130442480 Ki = 8000 nM T88547 CM04RF 130442572 Ki = 6900 nM T88547 CUD08L 134817200 Ki = 65.2 nM T88547 CZQS20 134828069 Ki = 5.7 nM T88547 CYB5V2 134828071 Ki = 5.1 nM T88547 CZ56GX 135423874 Ki = 743 nM T88547 CH96LU 135559170 Ki = 4000 nM T88547 C9C3LB 136056476 IC50 = 113 nM T88547 CN1I7A 137634153 Ki = 4200 nM T88547 CNH2K5 137639103 Ki = 2.3 nM T88547 C3Y8DJ 137643283 Ki = 2.6 nM T88547 CY56BC 137648624 Ki = 1.5 nM T88547 CU0OC3 137658890 Ki = 5.4 nM T88547 CC2DK4 137661600 Ki = 8.4 nM T88547 C1TQ2A 145953153 Ki = 6.5 nM T88547 CXEV63 145954849 Ki = 1418 nM T88547 CDGA65 145956728 Ki = 19 nM T88547 CZW93M 145979453 Ki = 99 nM T88547 CV43SZ 145980698 Ki = 57 nM T88547 C7H3GY 145986754 Ki = 38293 nM T88547 CC4KD9 145986903 Ki = 573 nM T88547 CS9R6C 145990153 Ki = 774 nM T88547 CC2G1V 146025727 Ki = 8800 nM T88547 CJA9T4 146597626 Ki = 15.85 nM T88547 C3D4UM 146597628 Ki > 10000 nM T88547 C7UHR0 146597630 Ki = 100 nM T88547 CCRS21 146597638 Ki > 10000 nM T88547 CM18OU 146597639 Ki = 2511.89 nM T88547 C42TIZ 146597651 Ki = 501.19 nM T88547 CL5PG8 146597666 Ki > 10000 nM T88547 C89YUC 146597677 Ki = 251.19 nM T88547 CU9G0O 146597678 Ki > 10000 nM T88547 C6TRC9 146641556 Ki = 316.23 nM T88547 C8I3YJ 146641558 Ki = 125.89 nM T88547 C3LBA0 146641564 Ki = 158.49 nM T88547 CFD4N9 146641568 Ki = 630.96 nM T88547 CP70WA 146641787 Ki = 251.19 nM T88547 C0WU5Y 146641788 Ki = 199.53 nM T88547 C10LOP 146641795 Ki > 10000 nM T88547 CG97ER 146709966 Ki = 3162.28 nM T88547 C6FX4M 147636204 Ki > 10000 nM T88547 CW4S2X 147652368 Ki > 10000 nM T88547 CF5B2L 147653864 Ki = 501.19 nM T88547 C5PNX8 148302367 Ki = 12.59 nM T88547 C2E5HK 149396365 Ki = 7.943 nM T88547 C9T0PS 153061504 Ki = 1000 nM T88547 CF7J3M 153287535 Ki = 50.12 nM T88547 C72MVW 153287537 Ki > 10000 nM T88547 CAF36V 153287539 Ki = 12.59 nM T88547 C1FA0K 153287541 Ki = 50.12 nM T88547 CEQ69Z 153287542 Ki = 39.81 nM T88547 C9A7SV 153287550 Ki > 10000 nM T88547 C91KST 153287551 Ki > 10000 nM T88547 C6P3SR 153287553 Ki = 501.19 nM T88547 C3G5CJ 153287557 Ki = 158.49 nM T88547 CW31CT 153287566 Ki = 162.18 nM T88547 CYP86E 153287567 Ki = 251.19 nM T88547 CS73ZC 153287568 Ki = 63.1 nM T88547 CV9G7Z 153287572 Ki = 1000 nM T88547 CO85KL 153287574 Ki = 316.23 nM T88547 CCD9N1 155512086 Ki = 1790 nM T88547 CTV8R1 155512151 Ki = 626 nM T88547 CV35ZN 155513505 Ki = 690 nM T88547 C0LR8C 155517675 Ki = 5.1 nM T88547 C4KWA1 155518665 Ki = 113 nM T88547 C0IHP6 155518770 Ki = 25.7 nM T88547 CUSA24 155519891 Ki = 39.81 nM T88547 C9W2NV 155525645 Ki = 31.62 nM T88547 CP76JX 155526977 Ki = 398.11 nM T88547 CQT9R0 155527577 Ki = 77.62 nM T88547 CQV19C 155528829 Ki = 55 nM T88547 CPA51T 155528865 Ki = 95 nM T88547 CMNU06 155529976 Ki = 20.89 nM T88547 CS2MF5 155532495 Ki = 251.19 nM T88547 CB79ZW 155536080 Ki = 125.89 nM T88547 C5IK2Y 155536631 Ki = 22 nM T88547 CR16NT 155540848 Ki = 63 nM T88547 CI7FN8 155545740 Ki = 21 nM T88547 CIA1C9 155547197 Ki = 63 nM T88547 CF7MQ8 155550094 Ki = 630.96 nM T88547 C8AGX6 155550691 Ki = 5.1 nM T88547 CI41QF 155552117 Ki = 1970 nM T88547 CJ92EA 155552895 Ki = 501.19 nM T88547 CKSZ39 155553997 Ki = 6.9 nM T88547 C04OFL 155554079 Ki = 7.2 nM T88547 CRU26E 155554287 Ki = 39.81 nM T88547 C6ZWX1 155554837 Ki = 16 nM T88547 CZ9U5N 155554849 Ki = 316.23 nM T88547 CC48RQ 155556295 Ki = 148 nM T88547 CBS89O 155556618 Ki = 1500 nM T88547 CQ7Y5M 155556668 Ki = 4.9 nM T88547 CJBX01 155557042 Ki = 125.89 nM T88547 C4J0ZI 155559223 Ki = 199.53 nM T88547 C13RCK 155561279 Ki = 70 nM T88547 CXYQ73 155561471 Ki = 63.1 nM T88547 CCOD50 155562467 Ki = 3570 nM T88547 C6YO5L 155562543 Ki = 43.65 nM T88547 CK9RN6 155563452 Ki = 24.55 nM T88547 CSM7V1 155564110 Ki = 30 nM T88547 CP9TR0 10324985 Ki = 480 nM T88547 CEA0P3 12233037 Ki = 0.67 nM T88547 CYZI29 12233038 Ki = 36.5 nM T88547 D00FUO 4416 Ki = 30 nM T88547 D00GSD 25107716 Ki > 5000 nM T88547 D00KIK 398369 Ki = 674 nM T88547 D00NQV 5041 Ki = 82.1 nM T88547 D00VHW 11152527 Ki = 2.5 nM T88547 D00VKV 62751 IC50 = 2060 nM T88547 D01HTH 60839 IC50 = 2535 nM T88547 D02BXG 398415 Ki = 3170 nM T88547 D02EHL 398376 Ki = 1730 nM T88547 D02WJT 7333 Ki = 15 nM T88547 D03LDH 10758200 Ki = 0.3 nM T88547 D03TDN 1342 Ki = 2720 nM T88547 D03TNT 5753 Ki = 35600 nM T88547 D04FBZ 5284595 IC50 = 48 nM T88547 D04JJL 14771671 IC50 = 245 nM T88547 D04JZJ 2838196 Ki = 370 nM T88547 D04LWD 11336800 Ki = 1.4 nM T88547 D04ZMS 11773145 Ki = 3.38 nM T88547 D05CGI 11245709 Ki = 1.4 nM T88547 D05EQG 5265 IC50 = 954.99 nM T88547 D06FUV 5311189 Ki = 234 nM T88547 D06RFW 13781937 IC50 = 270 nM T88547 D07AAZ 82553 IC50 = 1000 nM T88547 D07BAH 32893 Ki = 46400 nM T88547 D07OOI 3456 IC50 = 17 nM T88547 D07TKE 15723894 Ki = 3 nM T88547 D09CGH 188914 Ki = 1.26 nM T88547 D09NSH 10810249 Ki = 257.04 nM T88547 D09RPR 16737207 Ki > 10000 nM T88547 D09TDI 6472 Ki = 15.5 nM T88547 D0A0GU 44247568 Ki = 17 nM T88547 D0B3WX 5475158 IC50 = 181.97 nM T88547 D0C1LI 53378764 Ki = 2.83 nM T88547 D0E8FG 14952700 Ki = 2710 nM T88547 D0FF6S 16038374 IC50 > 10000 nM T88547 D0J1AE 10708590 Ki = 2.6 nM T88547 D0J6JT 1355 Ki = 6150 nM T88547 D0KL1P 10474335 Ki = 5.3 nM T88547 D0M4RW 5281878 IC50 = 14.79 nM T88547 D0N8WR 10390222 Ki = 92 nM T88547 D0O3GF 1220 Ki > 2427 nM T88547 D0P0XA 197060 Ki = 9310 nM T88547 D0Q5PC 6468 IC50 = 560 nM T88547 D0Q7FM 15443 Ki = 342 nM T88547 D0R5WX 11220953 Ki = 4.8 nM T88547 D0T1GZ 408731 Ki = 11.3 nM T88547 D0U3PC 398365 Ki = 9170 nM T88547 D0V4RP 1346 Ki = 11200 nM T88547 D0V5HV 4296 Ki = 1340 nM T88547 D0W2YN 2760172 Ki = 550 nM T88547 D0X4RC 7096 Ki = 11440 nM T88547 D0X7BG 4679312 Ki > 1000 nM T88547 D0Y3DR 608630 Ki = 2890 nM T97821 D0Y9EW 42611257 IC50 = 23 nM T97821 D04AHQ 71721540 IC50 = 39 nM T97821 D0Z1DH 10029385 IC50 > 20000 nM T97821 C31FHN 5330788 IC50 = 9970 nM T97821 CK2Q0Y 9972086 IC50 > 20000 nM T97821 CZV48E 9972935 IC50 = 16610 nM T97821 CU3D9T 9973794 IC50 > 20000 nM T97821 C6UJ3H 9995838 IC50 > 20000 nM T97821 CPZ34K 10002593 IC50 > 20000 nM T97821 C1XVD4 10049774 IC50 > 20000 nM T97821 C69VRQ 10064294 IC50 = 1310 nM T97821 C1TXC3 10094943 IC50 > 20000 nM T97821 CQP2T6 10321041 IC50 > 20000 nM T97821 CZV97C 10359218 IC50 = 2340 nM T97821 C8X2RY 10456042 IC50 = 8480 nM T97821 C30PKR 11248978 IC50 = 13400 nM T97821 CSXY78 11294864 IC50 > 20000 nM T97821 CPU9I3 11316975 IC50 > 20000 nM T97821 CQ8I4H 11328863 IC50 > 20000 nM T97821 CC96QB 11507696 IC50 > 20000 nM T97821 CYQ4O9 11723225 IC50 = 15940 nM T97821 CE9MU4 11740079 IC50 = 2810 nM T97821 CB5NF6 44408672 IC50 > 20000 nM T97821 CYG2F3 44408807 IC50 > 20000 nM T97821 CM54AI 44408849 IC50 = 15880 nM T97821 CN4X1A 44408884 IC50 = 4880 nM T97821 C3VRO9 44557921 IC50 > 10000 nM T97821 CLS29B 46872626 IC50 > 10000 nM T97821 CV63UL 67240318 IC50 > 10000 nM T97821 CM2J3B 131953483 IC50 = 5 nM T97821 CXC69T 137321158 IC50 = 457 nM T97821 C4P5VI 137631729 IC50 > 30000 nM T97821 C4N0LW 137631825 IC50 = 16.8 nM T97821 C0OWY3 137636794 IC50 = 22.6 nM T97821 C9SOI8 137644117 IC50 = 42.7 nM T97821 C23ACF 137644903 IC50 = 9.6 nM T97821 CQS67M 137644972 IC50 = 5.1 nM T97821 CIJK82 137647304 IC50 = 994.1 nM T97821 C97LQG 137647372 IC50 = 19.2 nM T97821 CJMW91 137649638 IC50 = 7.5 nM T97821 CF1H4X 137650051 IC50 = 143.7 nM T97821 CF2PV0 137655959 IC50 = 4.2 nM T97821 CHF87V 137657244 IC50 = 5.1 nM T97821 CN7J2A 137657347 IC50 = 12.1 nM T97821 C1W3PN 137661841 IC50 = 3.3 nM T97821 CM3UF7 137700779 IC50 > 10000 nM T97821 C2JI6T 138393294 IC50 = 4 nM T97821 CK90OA 138753620 IC50 = 2.1 nM T97821 CF57DG 146020550 IC50 = 4.2 nM T97821 CCO93U 154634893 IC50 = 4.4 nM T97821 C5DMK6 154634900 IC50 = 63.3 nM T97821 CVY7N6 154634909 IC50 = 3 nM T97821 C7YD9F 154634910 IC50 = 24.7 nM T97821 CE4V9P 154634911 IC50 = 4.5 nM T97821 C9CQ3T 154634913 IC50 = 2.3 nM T97821 CEC1D3 154634916 IC50 = 29 nM T97821 CGO62P 154634918 IC50 = 6.9 nM T97821 C41FIQ 154634920 IC50 = 3.8 nM T97821 C6XWC7 154634922 IC50 = 5.7 nM T97821 C2MD1Q 155513187 IC50 > 10000 nM T97821 C13KCF 155517164 IC50 = 85.7 nM T97821 CEZ4O1 155520166 IC50 = 1.9 nM T97821 CYZ16N 155526190 IC50 = 46.2 nM T97821 C6AGH4 155527315 IC50 = 983 nM T97821 CX0J3Y 155543780 IC50 = 54.3 nM T97821 CQXE36 155547334 IC50 = 53 nM T97821 C59PVM 155557441 IC50 = 8.9 nM T97821 CSA97I 155565690 IC50 = 3.3 nM T97821 C9QAE3 155566144 IC50 = 413.3 nM T97821 D00ERW 44444843 Ki > 8573 nM T97821 D06BDC 10361101 IC50 = 708 nM T97821 D0XB4P 447966 IC50 = 1400 nM T97821 D0Z5TQ 5924208 IC50 = 1890 nM T72595 D0I0DL 3689 IC50 = 29100 nM T72595 C63KYD 66637 IC50 = 15000 nM T72595 CD48TY 694463 IC50 = 68000 nM T72595 CD5RW2 1279398 IC50 = 2600 nM T72595 C5Z6NT 3113150 IC50 = 5400 nM T72595 CXF09D 4231127 EC50 = 2700 nM T72595 CN85UI 4235339 IC50 = 7000 nM T72595 C10ROQ 9972103 IC50 > 100000 nM T72595 C09KVR 9972180 IC50 > 100000 nM T72595 CGUQ10 10425979 IC50 > 100000 nM T72595 C4MCK2 10426105 IC50 > 100000 nM T72595 C3CID8 12045491 IC50 > 100000 nM T72595 C4Z0SE 12045492 IC50 > 100000 nM T72595 CN6RL1 12045493 IC50 > 100000 nM T72595 CJ0EZ4 12045494 IC50 > 100000 nM T72595 CM1S6P 12045495 IC50 > 100000 nM T72595 C13FGE 12045496 IC50 > 100000 nM T72595 CYL2J7 12045497 IC50 > 100000 nM T72595 CRB59C 12045498 IC50 = 51000 nM T72595 C27OQJ 12045832 IC50 > 100000 nM T72595 CI28HT 22432385 EC50 = 6600 nM T72595 CY0BC7 34924882 IC50 > 100000 nM T72595 CA72VD 44322229 IC50 = 12000 nM T72595 CQ21VN 44365962 IC50 > 100000 nM T72595 CDZ04W 44366039 IC50 > 100000 nM T72595 CCJD07 44366045 IC50 > 100000 nM T72595 C4BJ6F 44366056 IC50 > 100000 nM T72595 CR84AS 44366090 IC50 > 100000 nM T72595 C4DL5Q 44366109 IC50 > 100000 nM T72595 CRA24L 44366153 IC50 > 100000 nM T72595 C9CX5W 44366275 IC50 > 100000 nM T72595 CIC1G6 46861929 IC50 = 7100 nM T72595 C39CGI 56653056 IC50 = 50000 nM T72595 C4KWB0 56654447 EC50 = 37000 nM T72595 C7XPS1 66727815 IC50 = 2000 nM T72595 CN8M0L 90035858 EC50 = 13000 nM T72595 D06XGK 105074 EC50 = 83000 nM T72595 D09HXX 4787937 IC50 > 10000 nM T59190 D0E6XR 3062316 IC50 > 50000 nM T59190 D0E3TC 44259 IC50 = 216.8 nM T59190 D0I6VU 176167 IC50 = 8000 nM T59190 D0W3LI 153999 IC50 > 100000 nM T59190 D03BNU 59604787 IC50 > 10000 nM T59190 D0WS1V 448991 IC50 > 100000 nM T59190 D0CV8T 874670 EC50 = 3 nM T59190 D0Y7KX 71009752 EC50 = 2 nM T59190 D0YK9D 9956119 IC50 > 10000 nM T59190 D0R2TM 5287736 IC50 = 3500 nM T59190 C8OI7N 2290 IC50 = 3500 nM T59190 CLA43B 5327919 IC50 > 150000 nM T59190 CPDC54 5327920 IC50 > 150000 nM T59190 CCB9G3 5327921 IC50 > 150 nM T59190 CRTQ98 5327922 IC50 = 22000 nM T59190 CP20NQ 5327923 IC50 = 37000 nM T59190 CAO1N9 5327979 IC50 > 50000 nM T59190 C04EDX 9549298 EC50 = 3 nM T59190 C8J1OL 9826373 IC50 = 9000 nM T59190 C20NKA 9889351 IC50 = 4000 nM T59190 CV34AB 9958125 IC50 > 100000 nM T59190 C2W3AV 9995236 IC50 = 4000 nM T59190 C2UGV9 10030483 IC50 > 150000 nM T59190 C7YD1X 10048045 IC50 > 25000 nM T59190 CG7JO8 10099482 IC50 = 121000 nM T59190 C93LPQ 10099652 IC50 = 22500 nM T59190 C76TVG 10143584 IC50 > 10000 nM T59190 C7JP1A 10163439 IC50 = 4400 nM T59190 CJ0R2G 10187378 IC50 > 10000 nM T59190 C51SKM 10209082 IC50 = 6200 nM T59190 C7SFI1 10296883 IC50 = 5400 nM T59190 CAX9W2 10302405 IC50 = 5700 nM T59190 CEH41V 10392789 IC50 = 2800 nM T59190 C10PAC 10460251 IC50 = 39000 nM T59190 CX7S8N 10482293 IC50 = 1200 nM T59190 C76QGP 10506540 IC50 = 13000 nM T59190 CSR8Y5 10527068 IC50 = 44000 nM T59190 CDNP37 10530708 IC50 = 34000 nM T59190 C5EYJ3 10554684 IC50 > 150000 nM T59190 C71UIS 10555532 IC50 > 150000 nM T59190 CZ8UA9 10650891 IC50 > 5000 nM T59190 CJOU71 10671412 IC50 = 22000 nM T59190 CM5B6A 10673286 IC50 > 5000 nM T59190 CN9I6T 10768377 IC50 > 5000 nM T59190 CL8VH3 10768554 IC50 = 54000 nM T59190 C5YMK8 10769011 IC50 = 3100 nM T59190 C7HPA0 10864309 IC50 > 100000 nM T59190 C1DRE5 10884145 IC50 = 43 ug.mL-1 T59190 C1L4ZC 10940039 IC50 > 100000 nM T59190 CBOP58 11293798 Ki > 8000 nM T59190 C26BZX 11362471 Ki > 8000 nM T59190 CWXB93 11397177 Ki > 10000 nM T59190 C8DNQ2 11453012 IC50 = 4000 nM T59190 CK34LS 11632737 IC50 > 40000 nM T59190 CCX53Q 11729563 IC50 = 5000 nM T59190 CM10YB 11799388 IC50 = 55000 nM T59190 CA05OS 11972484 IC50 > 50000 nM T59190 C5RX1J 15096511 IC50 = 3500 nM T59190 C2BX8F 15297223 IC50 > 50000 nM T59190 CE04YW 15297224 IC50 > 50000 nM T59190 CFPW41 16007116 Ki > 8300 nM T59190 CGP40H 16784276 EC50 = 2 nM T59190 CVR9K4 22907281 IC50 = 9300 nM T59190 C0HRM6 22911602 IC50 = 7000 nM T59190 CUN67H 23366085 IC50 = 22000 nM T59190 CLG9Z8 23366090 IC50 > 50000 nM T59190 CW6OB1 23627212 IC50 > 100000 nM T59190 CKYB29 23644745 IC50 = 37000 nM T59190 CA3I4T 24753787 IC50 > 50000 nM T59190 C7YG1N 24759534 IC50 = 1900 nM T59190 C2UOE0 24766030 IC50 > 100000 nM T59190 CJUK39 24770517 IC50 > 50000 nM T59190 CM28WD 24825721 IC50 > 100000 nM T59190 CSW5V3 24865437 IC50 > 100 nM T59190 CJD12G 24943523 IC50 = 1210 nM T59190 CERG18 24970971 IC50 = 1590 nM T59190 CN2VT1 24970973 IC50 = 110 nM T59190 CPRA52 24970975 IC50 = 530 nM T59190 CLW80F 44160269 IC50 > 100000 nM T59190 CIX8V2 44251637 IC50 > 100000 nM T59190 CG1Z2B 44303442 IC50 = 42000 nM T59190 CNJ63O 44303517 IC50 = 9600 nM T59190 C8RJN7 44303745 IC50 > 50000 nM T59190 CTM59P 44308069 IC50 = 1200 nM T59190 CJ4WB9 44308383 IC50 = 12500 nM T59190 C1N6SL 44308409 IC50 > 150000 nM T59190 CO83HF 44308467 IC50 = 121000 nM T59190 CYTA85 44308468 IC50 > 150000 nM T59190 C3M4UP 44308469 IC50 > 150000 nM T59190 CY4K5F 44308490 IC50 = 3500 nM T59190 C7AG9Y 44308609 IC50 = 39000 nM T59190 CYN34A 44308610 IC50 = 3100 nM T59190 C79WUE 44308611 IC50 = 2800 nM T59190 CS63CK 44308612 IC50 = 34000 nM T59190 C47BNR 44310732 IC50 = 3500 nM T59190 C2ACB1 44310758 IC50 = 22000 nM T59190 CXVB19 44310795 IC50 = 37000 nM T59190 CD8OF2 44311036 IC50 > 150 nM T59190 C13TNU 44315122 IC50 = 56000 nM T59190 C3YN1R 44315123 IC50 > 150000 nM T59190 CPJ57U 44315124 IC50 = 37000 nM T59190 C9HA8T 44315171 IC50 = 16000 nM T59190 C2T3VN 44315184 IC50 > 50000 nM T59190 C3SP0H 44315423 IC50 > 50000 nM T59190 C8OAE9 44315457 IC50 > 150000 nM T59190 C3JS6X 44315503 IC50 = 37000 nM T59190 CEZ68T 44315545 IC50 > 150000 nM T59190 C5WL1F 44473009 IC50 > 100000 nM T59190 CEG1S5 44473011 IC50 > 100000 nM T59190 C46OMR 44473016 IC50 > 100000 nM T59190 CC95PQ 45375865 IC50 > 100000 nM T59190 CEOQ27 45375866 IC50 > 100000 nM T59190 CHC63L 45380888 IC50 = 33000 nM T59190 CO0C5D 45381091 IC50 = 14000 nM T59190 CICK85 45381093 IC50 = 30000 nM T59190 CEJ1F7 45381197 IC50 = 32000 nM T59190 CYKS07 45381199 IC50 = 12000 nM T59190 CSE95I 45381317 IC50 = 33000 nM T59190 C5S8MA 45485083 IC50 > 100000 nM T59190 CW42YX 45487634 IC50 > 100000 nM T59190 CQW97N 46846072 IC50 > 100000 nM T59190 CLS29B 46872626 IC50 > 10000 nM T59190 CHSF07 49806372 IC50 > 1000 nM T59190 C9L3XR 49838879 IC50 > 20000 nM T59190 CD4H3S 53354074 Ki > 5000 nM T59190 CI4DF2 54758213 IC50 = 28000 nM T59190 CA7JG9 54758215 IC50 = 13000 nM T59190 C5EYN1 56683794 IC50 = 17000 nM T59190 CBOD63 56835089 IC50 > 30000 nM T59190 CD6Y9Z 57395116 IC50 > 30000 nM T59190 C8W6IG 57395117 IC50 > 30000 nM T59190 CG7S0D 57396882 IC50 > 30000 nM T59190 CVK0G4 58056356 IC50 > 50000 nM T59190 COH41P 58325285 IC50 > 1000 nM T59190 CXJ63M 59603829 IC50 = 1800 nM T59190 CQEU96 59603842 IC50 = 40 nM T59190 CPAS93 60001348 EC50 = 1 nM T59190 CI7DY2 60965486 EC50 = 1 nM T59190 CV63UL 67240318 IC50 > 10000 nM T59190 C5DGR9 69036886 IC50 = 10000 nM T59190 C8T7ZP 70789255 IC50 = 74000 nM T59190 CH0B8N 70789756 IC50 > 30000 nM T59190 CX3H4C 71009783 EC50 = 1 nM T59190 C04WYL 71009786 EC50 = 10 nM T59190 CA3O6K 71552696 IC50 > 30000 nM T59190 C1NPL0 71552941 IC50 > 30000 nM T59190 CA4PS8 71552942 IC50 > 30000 nM T59190 CU60JG 71718528 IC50 > 50000 nM T59190 C7Q0AD 76286479 IC50 = 8500 nM T59190 CZF0N7 76287389 IC50 = 33000 nM T59190 CPG3A5 86302574 IC50 > 30000 nM T59190 C1HW4B 89735655 IC50 = 1100 nM T59190 CQ86OC 91799364 IC50 = 400 nM T59190 C0Y8ZK 91933875 IC50 > 1000 nM T59190 CX69OS 102340753 IC50 = 1000 nM T59190 CPI28L 102340754 IC50 = 3200 nM T59190 C4O0TP 118095304 IC50 = 2100 nM T59190 C15HSZ 118095336 IC50 = 600 nM T59190 CF5N1A 118095364 IC50 = 6200 nM T59190 CUY0N2 118095367 IC50 = 5400 nM T59190 CSJ30W 118095370 IC50 = 12700 nM T59190 C4VZJ0 118710696 IC50 = 9400 nM T59190 C3D2IF 118710697 IC50 = 11400 nM T59190 C2F7YV 118710698 IC50 = 8800 nM T59190 CT3QM1 118710699 IC50 = 12600 nM T59190 C2BDH1 118710701 IC50 = 5200 nM T59190 C3YV0I 118710702 IC50 = 2200 nM T59190 CA8JT9 118710703 IC50 = 2700 nM T59190 CXM0S5 118710704 IC50 = 3500 nM T59190 CX36UC 118710711 IC50 = 900 nM T59190 C5YEA1 118710712 IC50 = 900 nM T59190 CQ7MX1 118710713 IC50 = 700 nM T59190 CP3Z0R 118710714 IC50 = 28800 nM T59190 C1MNK2 118710718 IC50 = 5300 nM T59190 CTG50V 118710721 IC50 = 3700 nM T59190 C8ATN7 118710722 IC50 = 2900 nM T59190 CHS51O 118710723 IC50 = 300 nM T59190 C7ER0S 135566450 IC50 = 23.3 nM T59190 CUC08B 135566451 IC50 = 5.18 nM T59190 C6Q8IN 135839312 IC50 = 22 nM T59190 COM64Y 135928471 IC50 = 2.26 nM T59190 CYV4X9 135928472 IC50 = 5.6 nM T59190 C7N0LZ 135928473 IC50 = 290 nM T59190 CN0CT1 135928474 IC50 = 12400 nM T59190 CF94AE 135928475 IC50 = 5520 nM T59190 CN28FB 135928476 IC50 = 19000 nM T59190 CDO4A0 135928477 IC50 = 1510 nM T59190 CG0JQ5 135928478 IC50 = 55.5 nM T59190 CHX3L1 135928479 IC50 = 51.3 nM T59190 C1P9EO 135928480 IC50 = 31100 nM T59190 CIR82V 135928481 IC50 = 8800 nM T59190 CE2K9B 135928482 IC50 = 585 nM T59190 CMKZ30 135928483 IC50 = 1310 nM T59190 CR0M6N 135928484 IC50 = 27300 nM T59190 C4POF5 135928485 IC50 = 13600 nM T59190 CY47BR 135928486 IC50 = 11800 nM T59190 C8S3CO 135928487 IC50 = 8930 nM T59190 CQK06T 135928488 IC50 = 4080 nM T59190 CK9X8M 135928490 IC50 = 1070 nM T59190 CXFM96 136184114 IC50 = 6840 nM T59190 CDSW97 136184115 IC50 = 3020 nM T59190 CM32DP 136931811 IC50 = 1500 nM T59190 CM90WG 136931812 IC50 = 500 nM T59190 COQY54 136931814 IC50 < 100 nM T59190 CPL0W5 136931815 IC50 = 2500 nM T59190 CYED78 136931816 IC50 = 2900 nM T59190 CO3GA6 136931817 IC50 = 1400 nM T59190 CQEX28 136931818 IC50 = 720 nM T59190 C8DH9V 136931819 IC50 < 100 nM T59190 CI9ZH3 136951548 IC50 = 17400 nM T59190 CI1E8V 137634241 IC50 > 10000 nM T59190 CPH9E3 145967023 IC50 = 10 nM T59190 CK1D3Y 145979289 IC50 = 4300 nM T59190 CS14FQ 145979647 IC50 = 21300 nM T59190 C6FZH5 145981648 IC50 = 6500 nM T59190 CB72LP 145981790 IC50 < 100 nM T59190 C3U6KI 145988891 IC50 = 400 nM T59190 C68YQV 145989758 IC50 < 100 nM T59190 CVLR32 145991650 IC50 < 100 nM T59190 C47KPF 145991803 IC50 = 6200 nM T59190 C2MD1Q 155513187 IC50 > 10000 nM T59190 D00ERW 44444843 Ki > 8333 nM T59190 D02XHC 448912 IC50 > 100000 nM T59190 D06ZCX 10455969 IC50 = 8700 nM T59190 D07OAT 456214 IC50 > 100000 nM T59190 D0D6MH 11617559 IC50 > 24000 nM T59190 D0Q3KS 9957049 IC50 > 10000 nM T59190 D0TO6S 2396 IC50 = 5800 nM T59190 D0US9O 45275255 IC50 = 200 nM T72038 D02NDV 439357 IC50 = 50000000 nM T72038 CGRE80 23651530 IC50 = 5000000 nM T72038 C5PRE0 25022444 IC50 > 5000000 nM T72038 CSH54Y 44586823 IC50 > 5000000 nM T72038 C4ZAV3 44586861 IC50 > 5000000 nM T72038 CH6L3X 44586862 IC50 = 5000000 nM T72038 CTM7I3 44586863 IC50 > 5000000 nM T72038 C62VSK 44586864 IC50 = 5000000 nM T72038 CS9KL5 44586891 IC50 > 5000000 nM T72038 CJO0Y3 44586892 IC50 = 5000000 nM T72038 CGB59A 44586893 IC50 = 5000000 nM T72038 C1KTE2 44586894 IC50 = 2500000 nM T72038 CTZ16G 44586895 IC50 = 5000000 nM T72038 CY60FG 44586921 IC50 = 5000000 nM T72038 CUEA45 44586922 IC50 = 2500000 nM T72038 C0PC4W 44586923 IC50 = 2500000 nM T72038 CITZ01 44586924 IC50 = 2500000 nM T72038 C9Q6RH 44586925 IC50 = 2500000 nM T72038 CSVU02 44586950 IC50 > 5000000 nM T72038 CC5XY3 44586951 IC50 = 2500000 nM T72038 CL8WK0 44586952 IC50 = 2500000 nM T72038 CZ17UD 44586953 IC50 > 5000000 nM T72038 C1FYD6 44586954 IC50 = 5000000 nM T72038 CSM0P1 44586984 IC50 > 5000000 nM T72038 C5N4IP 44586985 IC50 = 300000 nM T72038 CBN67X 44586986 IC50 = 160000 nM T72038 CI4T9W 44586987 IC50 = 300000 nM T72038 C92USB 44586988 IC50 = 2500000 nM T72038 C1GJF9 44586989 IC50 = 300000 nM T72038 C5WJG0 44586990 IC50 > 5000000 nM T72038 CCU5M9 44587042 IC50 > 5000000 nM T72038 CL5M9D 44587043 IC50 = 160000 nM T72038 CQ4VC3 44587044 IC50 = 600000 nM T72038 CJGP86 44587045 IC50 = 2500000 nM T72038 CV7NL5 73348361 IC50 = 163000 nM T72038 CEG57V 145967201 EC50 = 17200 nM T72038 CEB75S 145967416 EC50 = 67700 nM T72038 CG6ZK8 145974460 EC50 = 18300 nM T72038 CDTL63 145975452 EC50 = 205000 nM T72038 C4TE7J 145976957 EC50 = 40700 nM T72038 D0K8XC 6134 IC50 = 800000 nM T39676 D00JAU 3749 IC50 > 500000 nM T39676 D00KHM 16362 IC50 > 500000 nM T39676 D00SEB 5388962 IC50 > 500000 nM T39676 D01AZG 5073 IC50 = 1600 nM T39676 D02DPA 2756 IC50 = 1200 nM T39676 D02KRS 2130 IC50 = 37800 nM T39676 D02PMO 60700 IC50 = 1300 nM T39676 D02YIZ 12560 IC50 > 500000 nM T39676 D03SKR 2803 IC50 = 33300 nM T39676 D05AHE 8226 IC50 > 250000 nM T39676 D05DVP 5717 IC50 = 1300 nM T39676 D05EAM 4735 IC50 = 2000 nM T39676 D05HSC 6000 IC50 = 9400 nM T39676 D05PHH 3447 IC50 = 500 nM T39676 D06NXY 5991 IC50 = 21100 nM T39676 D06ZUK 3696 IC50 = 10000 nM T39676 D07GRH 2749 IC50 > 500000 nM T39676 D07HOB 60838 IC50 = 7900 nM T39676 D08QCJ 5430 IC50 > 500000 nM T39676 D09FAZ 9444 IC50 > 500000 nM T39676 D0AV3G 3151 IC50 = 2300 nM T39676 D0AZ3C 5291 IC50 = 50 nM T39676 D0D7LA 4091 IC50 = 250000 nM T39676 D0D9FV 4601 IC50 = 65000 nM T39676 D0DK8V 2678 IC50 > 500000 nM T39676 D0DV3O 3241 IC50 = 1100 nM T39676 D0E6YQ 1935 IC50 = 1100 nM T39676 D0EP0C 5833 IC50 = 18600 nM T39676 D0F9GE 3108 IC50 = 26000 nM T39676 D0H3HM 60795 IC50 = 130000 nM T39676 D0IT2G 5743 IC50 > 500000 nM T39676 D0K0OZ 5702160 IC50 = 760 nM T39676 D0K7WK 4595 IC50 < 10 nM T39676 D0M4VM 5320 IC50 > 500000 nM T39676 D0M4YC 3114 IC50 = 66000 nM T39676 D0M7JT 216210 IC50 = 8100 nM T39676 D0N0ES 938 IC50 > 500000 nM T39676 D0N6RF 65999 IC50 = 17900 nM T39676 D0NR6S 3002977 IC50 = 17300 nM T39676 D0PQ3G 3440 IC50 > 500000 nM T39676 D0R1RS 3715 IC50 > 500000 nM T39676 D0R3JB 4212 IC50 = 400 nM T39676 D0T6XX 4679 IC50 = 2800 nM T39676 D0TG1H 3033 IC50 > 500000 nM T39676 D0TQ1G 5071 IC50 = 7300 nM T39676 D0U2OO 2477 IC50 = 1700 nM T39676 D0V3ZA 10531 IC50 = 2800 nM T39676 D0V4GY 9552079 IC50 = 700 nM T39676 D0V7CF 5362440 IC50 = 1900 nM T39676 D0W9LX 2585 IC50 = 92400 nM T39676 D0WV3U 4893 IC50 = 1600 nM T39676 D0X4RN 3676 IC50 > 500000 nM T39676 D0Z6UC 5358 IC50 = 6700 nM T39676 D0ZU9R 392622 IC50 = 80 nM T39676 D0Y6SQ 2536 IC50 = 2900 nM T39676 D0Y8AW 275196 IC50 = 34500 nM T39676 D0O2IE 4754 IC50 > 500000 nM T39676 D0QQ1J 2406 IC50 = 5200 nM T39676 D0Y2HR 2247 IC50 = 26400 nM T39676 CP4RM6 4486 IC50 = 650 nM T39676 C93BJO 5039 IC50 = 8300 nM T39676 C29SPL 5867 IC50 = 21400 nM T39676 CZA2C6 39764 IC50 = 1900 nM T39676 CLD6J9 441074 IC50 = 11200 nM T39676 CZLJ35 155554879 IC50 = 10000 nM T39676 D0P2HR 3510 IC50 = 5000 nM T14602 C5DP1O 1306479 IC50 = 7800 nM T14602 CZ7N5A 2283538 IC50 = 8900 nM T14602 CE5A7B 60162406 Ki > 30000 nM T14602 C30ZKJ 71561420 Ki > 50000 nM T14602 D0J1QT 44473100 Ki > 15000 nM T46216 D0PH9I 118693659 Ki = 2511.89 nM T46216 CL80QG 11820 IC50 = 14000 nM T46216 CG5O0H 638578 IC50 = 13700 nM T46216 C2M0SE 1511198 IC50 = 1258.93 nM T46216 CJK1F0 1511199 IC50 = 1584.89 nM T46216 CR3SF5 4907545 IC50 = 501.19 nM T46216 C3SC0O 16026457 IC50 = 204000 nM T46216 CG3PR6 52912222 IC50 > 31622.78 nM T46216 C0DNH5 53017606 IC50 = 48900 nM T46216 CUZR69 70680607 IC50 = 501.19 nM T46216 CDY89S 70680609 IC50 = 19900 nM T46216 CQ78NK 76310219 IC50 = 199.53 nM T46216 CM4J8Q 76317442 IC50 = 316.23 nM T46216 CM7TH3 76328466 IC50 = 630.96 nM T46216 C0T5NK 76335637 IC50 = 1000 nM T46216 CYF7O2 91668539 IC50 = 12.59 nM T46216 C2JXG5 91668540 IC50 = 15.85 nM T46216 CZ0H2Y 91668542 IC50 = 199.53 nM T46216 C9WB3G 95828281 IC50 > 20000 nM T46216 CIX5V3 113222223 IC50 > 50118.72 nM T46216 CB5O8P 115579930 IC50 > 50118.72 nM T46216 CVA75B 115611029 IC50 > 50118.72 nM T46216 CYX7T2 117072549 IC50 = 75 nM T46216 C87ZPY 118796358 IC50 = 19 nM T46216 CRF4G8 118796361 IC50 = 21 nM T46216 CWS6Y5 118796362 IC50 = 9338 nM T46216 CF9J8E 118918705 IC50 = 170 nM T46216 CA3Z8O 118918714 IC50 = 910 nM T46216 C8GLJ3 118918720 IC50 = 2500 nM T46216 C2ZY3U 118932975 IC50 = 2700 nM T46216 CC14FI 118933132 IC50 = 310 nM T46216 CGO91Y 118933136 IC50 = 890 nM T46216 C8AZ4C 119081691 IC50 = 1400 nM T46216 CUWX94 119081692 IC50 = 230 nM T46216 C9MQF0 119098887 IC50 = 57 nM T46216 C0QX4D 119098889 IC50 = 30 nM T46216 CB83MK 121271792 IC50 = 730 nM T46216 CP1NH2 121277975 IC50 > 20000 nM T46216 C3GD2W 121335190 IC50 = 160 nM T46216 C81OYL 121335218 IC50 = 18000 nM T46216 C83RUE 121335260 IC50 = 750 nM T46216 CECP26 121335281 IC50 = 290 nM T46216 C1HR3M 121335283 IC50 = 9500 nM T46216 C2EP5S 121335312 IC50 = 2200 nM T46216 CNW25A 121338193 IC50 = 11000 nM T46216 C5JYP8 121338332 IC50 = 6900 nM T46216 C5ML2V 121338401 IC50 = 8500 nM T46216 C3JMB8 121338437 IC50 = 5000 nM T46216 CF25LT 121338490 IC50 = 2400 nM T46216 C5US9K 121338530 IC50 = 17800 nM T46216 CMF5D4 121338574 IC50 > 20000 nM T46216 C0VF7X 121338589 IC50 = 11400 nM T46216 CQ30XW 121342392 IC50 = 1400 nM T46216 CNM34X 121342393 IC50 = 620 nM T46216 CXI0K8 121342398 IC50 = 960 nM T46216 C9O4RD 121342404 IC50 = 1600 nM T46216 CJMF61 121342523 IC50 = 3000 nM T46216 CQKU78 121342528 IC50 = 2200 nM T46216 CDH8M4 121373418 IC50 > 20000 nM T46216 C47QXT 121376807 IC50 > 20000 nM T46216 C38ERO 121472643 IC50 > 50118.72 nM T46216 C1OIJ9 121476448 IC50 > 50118.72 nM T46216 C5B4TZ 123773279 EC50 = 320 nM T46216 CG9S7A 126961735 IC50 = 7943.28 nM T46216 CJR0V7 127025419 IC50 = 79.43 nM T46216 CZ93IW 127025420 IC50 = 7.943 nM T46216 C5FV9L 127025697 IC50 = 10 nM T46216 C8N5UA 127025979 IC50 = 39.81 nM T46216 C7M2GL 127025980 IC50 = 3981.07 nM T46216 C2LYR4 127025981 IC50 = 5011.87 nM T46216 C8GLF2 127025982 IC50 = 125.89 nM T46216 CMG7C1 127026579 IC50 = 23700 nM T46216 C57IHP 127026582 IC50 = 17900 nM T46216 CF9QV5 127026591 IC50 > 50000 nM T46216 C4MY5E 127026593 IC50 = 3162.28 nM T46216 C7OQT2 127026594 IC50 = 39.81 nM T46216 C62OFC 127026595 IC50 = 12.59 nM T46216 C0C1HZ 127028091 IC50 = 1400 nM T46216 C3R8FQ 127038798 IC50 = 125.89 nM T46216 CBNZ13 127040778 IC50 = 2511.89 nM T46216 CTA9I1 127042046 IC50 = 501.19 nM T46216 CGA71L 127048256 IC50 = 134 nM T46216 CH6T5J 127048257 IC50 = 507 nM T46216 C60SZQ 127048258 IC50 = 134 nM T46216 C5AV7U 127049278 IC50 = 1147 nM T46216 C50BMV 127049279 IC50 = 54 nM T46216 CTFY41 127049280 IC50 = 656 nM T46216 CVE71A 127049281 IC50 = 195 nM T46216 C73TND 127049282 IC50 = 468 nM T46216 C2VC3L 127050405 IC50 = 9 nM T46216 CWFM08 127050492 IC50 = 470 nM T46216 CTF4N2 127051087 IC50 = 37 nM T46216 CLSZ47 127051725 IC50 = 37 nM T46216 CMY93U 127051726 IC50 = 250 nM T46216 CY8V1A 127051727 IC50 = 128 nM T46216 CXZT48 127052023 IC50 = 134 nM T46216 CGM6W4 128963618 IC50 = 4400 nM T46216 CA0P5D 131953422 IC50 = 1995.26 nM T46216 CK0B6N 131985884 IC50 = 220 nM T46216 COE15M 132166121 IC50 = 1400 nM T46216 C7KUC2 132176755 IC50 = 7600 nM T46216 CGDN94 132275066 IC50 > 20000 nM T46216 CHL8K4 132941768 IC50 = 31622.78 nM T46216 CS7WX6 134821995 IC50 = 1500 nM T46216 CIAG86 135394452 IC50 = 1600 nM T46216 CD4NE1 137633137 IC50 = 9300 nM T46216 C5I9TL 137634095 IC50 = 2511.89 nM T46216 CYU6T2 137634563 IC50 = 5700 nM T46216 C2IHE8 137635251 IC50 > 50118.72 nM T46216 CQT3A9 137636309 IC50 > 20000 nM T46216 CV1EP8 137639742 IC50 = 9800 nM T46216 CL4FK6 137641456 IC50 > 20000 nM T46216 CZXP42 137644405 IC50 = 3500 nM T46216 CULX38 137646779 IC50 = 31622.78 nM T46216 CGX65O 137647885 IC50 = 5800 nM T46216 CM6S0X 137650255 IC50 = 2600 nM T46216 CC34KQ 137650533 IC50 = 420 nM T46216 C1MA2K 137651137 IC50 = 1500 nM T46216 C5Y0DH 137651263 IC50 = 3500 nM T46216 C6SKI2 137651884 IC50 = 3300 nM T46216 CV7G1I 137654127 IC50 = 1258.93 nM T46216 C7L6MV 137655172 IC50 = 6100 nM T46216 C1N7LY 137658279 IC50 = 1700 nM T46216 CQ6XB7 139030526 IC50 > 50118.72 nM T46216 C8ZQ2U 141736359 IC50 > 20000 nM T46216 C5VNM4 141736367 IC50 > 20000 nM T46216 C96NCH 145950955 IC50 > 20000 nM T46216 C3ZV1O 145952497 IC50 > 20000 nM T46216 CTE74G 145954441 IC50 > 20000 nM T46216 CN5YO3 145957310 IC50 > 20000 nM T46216 C7C5WL 145958595 IC50 > 20000 nM T46216 C2KC6G 155510588 IC50 = 730 nM T46216 C30COX 155514594 IC50 = 1600 nM T46216 CX5W9H 155515117 IC50 = 860 nM T46216 C8HK5X 155518008 IC50 = 2400 nM T46216 CFVU05 155519921 IC50 = 880 nM T46216 CN6YC5 155520197 IC50 = 967 nM T46216 CKD9U4 155526975 IC50 = 2100 nM T46216 CVY04U 155527380 IC50 = 2000 nM T46216 CL9VB6 155531262 IC50 = 1000 nM T46216 CQN6G3 155532286 IC50 = 1800 nM T46216 C0QV9U 155534567 IC50 = 890 nM T46216 CG9A4B 155540734 IC50 = 480 nM T46216 C62EMT 155540785 IC50 = 1000 nM T46216 C7VRN8 155541456 IC50 = 1700 nM T46216 C1Q6DU 155542223 IC50 = 557 nM T46216 C2JBP0 155543000 IC50 = 465 nM T46216 CW26QE 155544106 IC50 = 262 nM T46216 CV69DA 155544211 IC50 = 438 nM T46216 CW0S4Z 155545163 IC50 = 827 nM T46216 CEB37H 155547641 IC50 = 763 nM T46216 C6A3QM 155550203 IC50 = 3012 nM T46216 C0TBA1 155550442 IC50 = 7208 nM T46216 CF8V4I 155550513 IC50 = 1502 nM T46216 C56PTX 155550768 IC50 = 652 nM T46216 C74RSJ 155551627 IC50 = 802 nM T46216 C4PN0R 155554522 IC50 = 35 nM T46216 CLF6E3 155555073 IC50 = 2326 nM T46216 C1O9FC 155557989 IC50 = 103 nM T46216 CCH31L 155557990 IC50 = 7410 nM T46216 C3FL1B 155560778 IC50 = 1021 nM T46216 CI1ZU8 155561055 IC50 = 1700 nM T46216 C92XZO 155561955 IC50 = 930 nM T46216 C5NU8A 155564453 IC50 = 900 nM T46216 CD8WQ2 155565973 IC50 = 840 nM T46216 D03XXT 72201027 IC50 > 20000 nM T46216 D07ALG 72943187 IC50 = 160 nM T46216 D08LXU 91827372 IC50 = 3300 nM T46216 D0N5BI 91668541 IC50 = 50.12 nM T46216 D0O6XT 91827373 IC50 = 4400 nM T46216 D0T3WL 73010930 IC50 > 50000 nM T85540 CWJ0U1 5312 IC50 = 4500 nM T85540 C06WZQ 222878 IC50 = 480 nM T85540 COS62U 245007 IC50 > 100000 nM T85540 C0MHV8 252439 IC50 = 1900 nM T85540 C2OS3W 2238068 IC50 > 100000 nM T85540 CEQ4V8 2723716 IC50 > 100000 nM T85540 CCYF63 9942424 IC50 = 630.96 nM T85540 CW01ZQ 22581416 IC50 = 71900 nM T85540 C75LNS 22581449 IC50 = 52800 nM T85540 CF47JU 25138011 IC50 = 30 nM T85540 C7X3WA 28330466 IC50 > 100000 nM T85540 CL3HT1 71449736 IC50 = 42000 nM T85540 CJH86V 71451542 IC50 > 100000 nM T85540 CH38AO 71453382 IC50 > 100000 nM T85540 C2U4AQ 71458738 IC50 = 1100 nM T85540 C68RKH 76310231 IC50 = 26000 nM T85540 CO1EN3 76317452 IC50 = 190 nM T85540 CT5FZ8 76321184 IC50 = 35000 nM T85540 C6XRT0 76321186 IC50 = 8500 nM T85540 CKB5O9 76328366 IC50 = 37000 nM T85540 CUNK03 76335652 IC50 = 21000 nM T85540 CX23ZP 78426670 IC50 = 250 nM T85540 CMR52S 78426698 IC50 = 14 nM T85540 CKXW73 78427224 IC50 < 250 nM T85540 C63ATV 81750201 IC50 = 100 nM T85540 CRQ51Z 86346639 IC50 < 100 nM T85540 C83TUW 89825693 IC50 = 125.89 nM T85540 CT46KN 90094283 IC50 < 1000 nM T85540 CG4BZ9 90094442 IC50 < 1000 nM T85540 C2NA5I 91801131 IC50 = 12589.25 nM T85540 CP3DK0 96607511 IC50 = 12 nM T85540 C85UGZ 96608360 IC50 = 1700 nM T85540 CCZ4Q9 96617507 IC50 = 122 nM T85540 C10RDJ 101882871 IC50 = 1995.26 nM T85540 CY87WL 112499933 IC50 = 6800 nM T85540 C4FPD3 112726150 IC50 > 100000 nM T85540 C7TBE9 118908379 IC50 = 65.5 nM T85540 CJVK69 119081409 IC50 = 55 nM T85540 CRM93S 122181583 IC50 = 28900 nM T85540 C75JVN 122191451 IC50 = 6309.57 nM T85540 C3YX7W 122191453 IC50 = 10000 nM T85540 C3IBR8 122191455 IC50 = 5011.87 nM T85540 C59KNQ 122191457 IC50 = 7943.28 nM T85540 CM5X8J 122191459 IC50 = 7943.28 nM T85540 C7ASR0 122191460 IC50 = 10000 nM T85540 CRI6J4 122191461 IC50 = 3981.07 nM T85540 CAS4H6 122191462 IC50 = 5011.87 nM T85540 C9J6LX 122191463 IC50 = 6309.57 nM T85540 C75NJO 122191464 IC50 = 3981.07 nM T85540 C50VYK 122191465 IC50 = 3981.07 nM T85540 CSKY20 122191466 IC50 = 3162.28 nM T85540 CS3L8H 122191467 IC50 = 630.96 nM T85540 CZ2NV1 122191468 IC50 = 2511.89 nM T85540 CYTW93 122191469 IC50 = 6309.57 nM T85540 CZV45H 122191470 IC50 = 3981.07 nM T85540 CF6I2N 122191471 IC50 = 6309.57 nM T85540 CZU02B 122191472 IC50 = 1258.93 nM T85540 CE27AS 122191473 IC50 = 3162.28 nM T85540 CAJ28B 122191475 IC50 = 6309.57 nM T85540 C36PDK 122191476 IC50 = 1995.26 nM T85540 CQ04FW 122191477 IC50 = 2511.89 nM T85540 C12OHA 122191478 IC50 = 3981.07 nM T85540 CL2K0J 122191479 IC50 = 5011.87 nM T85540 CT6HG3 122191480 IC50 = 10000 nM T85540 CK7LD6 122191481 IC50 = 7943.28 nM T85540 CMJ72N 122191482 IC50 = 5011.87 nM T85540 C6H2YQ 122383780 IC50 = 178000 nM T85540 CT2UZ4 125377518 IC50 > 100000 nM T85540 C2FPM6 127031758 IC50 = 2000 nM T85540 C7W8TS 127031759 IC50 = 30 nM T85540 CMJE83 127031760 IC50 = 60 nM T85540 C2Z6CV 135567105 IC50 = 331 nM T85540 CIW61V 135567106 IC50 = 2000 nM T85540 CNZ8K9 135567107 IC50 = 830 nM T85540 CL9ZD4 135567108 IC50 = 78 nM T85540 CJM4Z2 135567109 IC50 = 340 nM T85540 CDY98J 135567110 IC50 = 67 nM T85540 C1VAI3 135567112 IC50 = 23 nM T85540 CWI0N7 135567114 IC50 = 9400 nM T85540 C8LFY7 135567115 IC50 = 51 nM T85540 C5E0ZN 135567116 IC50 = 440 nM T85540 CO1F4A 135567128 IC50 = 63.1 nM T85540 CWCY64 136048725 IC50 = 8400 nM T85540 CE1SW8 136053677 IC50 = 79.43 nM T85540 CMW30T 136053680 IC50 = 125.89 nM T85540 C6IJ5M 136053683 IC50 = 125.89 nM T85540 CNY5T7 136053684 IC50 = 199.53 nM T85540 C2V6MX 136644692 IC50 = 31622.78 nM T85540 CF5XJ1 137146154 IC50 = 7300 nM T85540 CK8DR7 137174994 IC50 = 150 nM T85540 CA6DH2 137174995 IC50 = 342 nM T85540 CLDH80 137174999 IC50 = 80 nM T85540 CR37AY 137175000 IC50 = 136 nM T85540 C1J3YB 137175001 IC50 = 76 nM T85540 CGAS95 137175002 IC50 = 64 nM T85540 CS5C6F 137175084 IC50 = 103400 nM T85540 C7PZ2T 137175085 IC50 = 730 nM T85540 C1B5CK 137175086 IC50 = 1300 nM T85540 CWV4Y6 137175087 IC50 > 100000 nM T85540 C9XOV5 137175088 IC50 = 88000 nM T85540 C34LUV 137175094 IC50 = 65 nM T85540 CSWN28 137175120 IC50 = 126 nM T85540 C23GYQ 137175121 IC50 = 54 nM T85540 C8Y2PR 137175122 IC50 = 70 nM T85540 C7GUC3 137175140 IC50 = 21 nM T85540 CBD1Q8 137175175 IC50 = 50 nM T85540 CEL6B1 137175176 IC50 = 57 nM T85540 C7SC6T 137175177 IC50 = 52 nM T85540 CPU73A 137175178 IC50 = 34 nM T85540 CFJ76N 137175179 IC50 = 119 nM T85540 CA89LW 137175180 IC50 = 142 nM T85540 C5GV3Q 137175209 IC50 = 50 nM T85540 C93YUK 137175210 IC50 = 46 nM T85540 CB2XV7 137175225 IC50 = 111000 nM T85540 C0XN8Y 137175239 IC50 = 8400 nM T85540 CI4D3P 137175249 IC50 = 41 nM T85540 CTVD83 137175250 IC50 = 21 nM T85540 C80LCT 137175251 IC50 = 22 nM T85540 CKQ1I2 137175252 IC50 = 23 nM T85540 C1YGB9 137175253 IC50 = 41 nM T85540 C5OZR6 137175260 IC50 = 32 nM T85540 CIKW02 137175261 IC50 = 24 nM T85540 C7J1RC 138393333 IC50 = 163 nM T85540 CYG29R 138393334 IC50 = 48 nM T85540 CNG82D 138393336 IC50 = 123 nM T85540 CPFZ83 138393339 IC50 = 132 nM T85540 C1ANF3 138518187 IC50 = 170 nM T85540 CXV31U 138753208 IC50 = 246 nM T85540 C41KVR 138753209 IC50 = 53 nM T85540 CIQJ26 138753211 IC50 = 14 nM T85540 CARJ34 138753212 IC50 = 202 nM T85540 CEQD63 155510449 IC50 = 96 nM T85540 CCB54Y 155510907 IC50 = 214 nM T85540 CAMR98 155512849 IC50 = 549 nM T85540 C9TWS3 155514456 IC50 = 35 nM T85540 C7XNM9 155518054 IC50 = 856 nM T85540 C4M1EO 155519111 IC50 = 96 nM T85540 CRT5Z2 155525082 IC50 = 566 nM T85540 CMB9N3 155530704 IC50 = 470 nM T85540 C2HN9G 155536799 IC50 = 213 nM T85540 C7VX3Y 155538517 IC50 = 156 nM T85540 CP8K5E 155540290 IC50 = 38 nM T85540 C7LFH3 155540572 IC50 = 377 nM T85540 CTF1K9 155542268 IC50 = 63 nM T85540 C7EG9J 155543678 IC50 = 313 nM T85540 C3M0TR 155546359 IC50 = 571 nM T85540 CIM7D4 155548682 IC50 = 5.84 nM T85540 C1CNK5 155549007 IC50 = 86 nM T85540 CX9OP1 155550806 IC50 = 113 nM T85540 CFR06L 155551969 IC50 = 6.24 nM T85540 C48ANL 155557731 IC50 = 54 nM T85540 C4MU5J 155558505 IC50 = 81 nM T85540 CTDM51 155558717 IC50 = 79 nM T85540 CPOM30 155560356 IC50 = 59 nM T85540 CA9T8I 155563296 IC50 = 896 nM T85540 CGCN43 155567831 IC50 = 108 nM T85540 C3SQ4A 155569285 IC50 = 30 nM T85540 D07IOY 10365 IC50 = 501.19 nM T85540 D08IZY 3080614 IC50 = 7943.28 nM T85540 D0B2WZ 15331 IC50 > 100000 nM T85540 D0X5US 459617 IC50 = 25000 nM T30563 C3TVL7 23501721 IC50 = 3060 nM T30563 CJMZ37 25174150 IC50 = 143 nM T30563 CV3TA6 25192021 IC50 = 628 nM T30563 C7A8UE 25192471 IC50 = 194 nM T30563 D0V3ZG 25192022 IC50 = 164 nM T36423 D0ZM5O 9884366 IC50 > 1000 nM T36423 CO9VA3 9820671 IC50 > 1000 nM T36423 C7SMT0 9908904 IC50 > 1000 nM T36423 CAM63X 42618195 IC50 > 1000 nM T36423 C8K4UF 42618197 IC50 > 1000 nM T81183 D01AZG 5073 Ki = 0.69 nM T81183 D01UXC 2249 IC50 = 230 nM T81183 D03SKR 2803 EC50 = 290 nM T81183 D05DVP 5717 IC50 > 10000 nM T81183 D06XZR 27400 Ki = 75 nM T81183 D07MOX 439260 Ki = 2600 nM T81183 D0AE3X 2435 Ki = 1800 nM T81183 D0D1AL 3559 Ki = 5.7 nM T81183 D0E9PK 4810 Ki > 30000 nM T81183 D0H7KF 5002 Ki = 4.5 nM T81183 D0I8FI 3779 EC50 = 1.5 nM T81183 D0MT0M 2216 EC50 = 180 nM T81183 D0R1JV 60854 Ki = 1.9 nM T81183 D0R6BI 3341 Ki = 151.36 nM T81183 D0T6QX 5736 Ki = 3.4 nM T81183 D0T7OW 681 Ki = 2511.89 nM T81183 D0V4QS 135398745 Ki = 7.3 nM T81183 D0WV3U 4893 Ki = 0.054 nM T81183 D0X6BV 6918314 IC50 = 1980 nM T81183 D0Z1RV 135398737 Ki = 3.7 nM T81183 D07WHS 5312115 EC50 > 1000000 nM T81183 D0F2ML 68602 EC50 = 1165 nM T81183 D07YLK 4350931 Ki = 11 nM T81183 D01WJZ 60820 Ki = 1.3 nM T81183 D02FNU 56971 IC50 = 500 nM T81183 D06DZI 107780 Ki < 1000 nM T81183 D08SOF 5405 IC50 = 2340 nM T81183 D0BC6Q 9837551 Ki = 470 nM T81183 D0EE6L 3038495 Ki = 5 nM T81183 D0K0DB 6604887 Ki = 180 nM T81183 D0K9JP 9928332 Ki > 1000 nM T81183 D0O9EM 208928 Ki > 10000 nM T81183 D0OS6O 60149 Ki = 1.8 nM T81183 D0W7IR 9887884 Ki = 3900 nM T81183 D0Y1PG 9841972 EC50 = 5600 nM T81183 D0ZG9N 132337 Ki > 10000 nM T81183 C4JQ7T 2068 Ki > 100000 nM T81183 CZUI83 2769 IC50 = 30 nM T81183 CK1JY9 3106 Ki = 1995.26 nM T81183 C0H8GR 3191 IC50 = 183 nM T81183 C2H1VA 131829 Ki = 1100 nM T81183 CZL87W 133999 IC50 > 10000 nM T81183 CF4V5Q 185076 Ki = 1400 nM T81183 C64CQL 385013 Ki = 76 nM T81183 C1VE3T 386224 Ki = 79 nM T81183 CT3UV7 444005 IC50 > 1000 nM T81183 CJ30IQ 1248739 Ki = 260 nM T81183 C64CZV 3038494 Ki = 5 nM T81183 C54QJC 3086247 Ki = 2400 nM T81183 CWNZ35 6469693 Ki = 98 nM T81183 CJTQ40 6469918 Ki = 60 nM T81183 C9R7NM 9104271 IC50 = 88 nM T81183 CHD32K 9794524 Ki > 28000 nM T81183 C4K7ZJ 9795515 Ki = 4200 nM T81183 CLUT03 9799123 IC50 = 1257 nM T81183 CCSN93 9800737 IC50 = 1000 nM T81183 CX7I8J 9802187 Ki = 16 nM T81183 CX3U7N 9813501 Ki = 430 nM T81183 CJM0W8 9816863 Ki = 2300 nM T81183 C45QPU 9820163 Ki = 1 nM T81183 C95BXW 9823464 IC50 = 100 nM T81183 CJ8LT7 9848518 IC50 > 10000 nM T81183 CB31LS 9855978 Ki = 1200 nM T81183 CTUM52 9856417 Ki = 1700 nM T81183 C3YSQ5 9859238 Ki = 5100 nM T81183 CQ2L0J 9859437 Ki = 16000 nM T81183 C7EZ2L 9859861 Ki > 10000 nM T81183 C5WYN4 9865858 Ki = 53 nM T81183 C3GMU5 9868889 Ki = 1.2 nM T81183 CA87LO 9869262 Ki = 56.23 nM T81183 CT2C6K 9870702 IC50 > 10000 nM T81183 CK76MQ 9872238 Ki = 0.4 nM T81183 CYSB08 9878065 Ki = 730 nM T81183 CPI8G9 9881158 Ki = 1500 nM T81183 C3DB5H 9884781 Ki = 967 nM T81183 C9GB2M 9888555 Ki = 15 nM T81183 CDLB96 9889149 IC50 = 100 nM T81183 C1ANB8 9889726 Ki = 1.99 nM T81183 C6CZ3G 9906777 IC50 > 10000 nM T81183 CO7BK6 9909648 Ki = 38 nM T81183 CQ3L1X 9921302 Ki = 670 nM T81183 CJ46NU 9921303 Ki = 490 nM T81183 CBE1Y9 9921863 Ki = 3300 nM T81183 CH5D3J 9928343 IC50 > 10000 nM T81183 C5V0UE 9933975 Ki = 41.1 nM T81183 C5E7KC 9943680 Ki = 3200 nM T81183 C1K8WB 9951233 Ki = 2003 nM T81183 C4I7UJ 9964754 Ki = 1000 nM T81183 CQIU94 9978693 IC50 = 700 nM T81183 CC6M7Z 9980998 Ki > 10000 nM T81183 C2C1XS 10042602 Ki = 67.61 nM T81183 C2JZL1 10048222 IC50 > 1000 nM T81183 C4GHO2 10053476 Ki > 1000 nM T81183 CJXQ40 10092819 Ki = 8.6 nM T81183 CRS5B6 10176999 Ki = 2100 nM T81183 CQ8HX2 10198135 Ki = 8400 nM T81183 C6S2RA 10198552 Ki = 130 nM T81183 CC2KV3 10214826 Ki > 100000 nM T81183 CE9Y8J 10276451 Ki = 370 nM T81183 C9LWG3 10369004 IC50 = 59 nM T81183 CS2DN8 10376336 EC50 = 12692 nM T81183 C69KIB 10385855 IC50 > 10000 nM T81183 C4UN0A 10436653 Ki = 15 nM T81183 C8KD1B 10438027 Ki = 300 nM T81183 CO7IV6 10450593 Ki = 8 nM T81183 CIA16B 10457445 Ki = 389.05 nM T81183 C26KCR 10475231 Ki = 100 nM T81183 CPI5M7 10476504 Ki = 26 nM T81183 C48BRW 10546334 Ki = 93.33 nM T81183 CBOS60 10548781 Ki = 38 nM T81183 C6O9CB 10572092 Ki > 500 nM T81183 C1DXO0 10609673 Ki = 6600 nM T81183 CFC42Z 10664759 Ki = 47 nM T81183 CI0GO3 10666853 Ki = 234 nM T81183 CTSY18 10682720 Ki = 16000 nM T81183 C3LDA1 10690393 Ki = 44 nM T81183 CP0B6F 10691211 Ki = 33 nM T81183 CYRG83 10714368 Ki = 94 nM T81183 C0USP7 10718592 Ki = 1.7 nM T81183 C3OCI1 10731942 Ki = 16 nM T81183 C4EZS5 10736855 Ki = 132 nM T81183 C5Z3JE 10737897 Ki = 2.3 nM T81183 CIZ05K 10761543 Ki = 74 nM T81183 C9HWI2 10783359 Ki = 18 nM T81183 CG12BP 10784327 Ki > 500 nM T81183 C3P2VZ 10785265 Ki = 23 nM T81183 C1P4GW 10785266 Ki = 20 nM T81183 C81PIH 10807090 Ki = 117 nM T81183 CD92GV 10832838 Ki = 35 nM T81183 C9A8KN 10862425 Ki = 19 nM T81183 CMV36C 10884046 Ki = 48 nM T81183 CRI50E 10885636 IC50 = 1100 nM T81183 CX65PW 10907460 IC50 = 993 nM T81183 CU09AV 10937901 IC50 = 1330 nM T81183 CSLT97 10949380 IC50 = 4920 nM T81183 C2HP7F 10981761 IC50 = 4250 nM T81183 CJC9K4 11005810 IC50 = 417 nM T81183 CB7N1P 11035765 IC50 = 174 nM T81183 CFJG64 11059058 IC50 = 1340 nM T81183 CG41BK 11071079 IC50 = 1640 nM T81183 C7DE0U 11113605 IC50 = 1170 nM T81183 C75WKP 11176199 IC50 = 45 nM T81183 C8JW3Z 11260311 Ki = 140 nM T81183 C4S2VF 11277147 Ki > 1000 nM T81183 CJS9C0 11304851 IC50 = 1000 nM T81183 CN63TR 11504230 Ki = 2.5 nM T81183 C16TWK 11508052 IC50 > 10000 nM T81183 C59SCV 11516033 Ki = 61 nM T81183 CW68BJ 11518143 IC50 = 1000 nM T81183 CXWO08 11522273 IC50 > 10000 nM T81183 CY5I0U 11559581 Ki = 380 nM T81183 CNH1K4 11568826 Ki = 13.7 nM T81183 C8CU1X 11581237 Ki = 64 nM T81183 C4L7TV 11662592 Ki = 118.1 nM T81183 CTK8R9 11678172 Ki = 80 nM T81183 CEQ6W7 11694810 Ki > 1000 nM T81183 C1W8NR 11696910 Ki = 190 nM T81183 CKT7L2 11698732 Ki = 2.64 nM T81183 CB4H2O 11699469 Ki = 8.4 nM T81183 CJL61W 11706497 Ki = 480 nM T81183 CGO56C 11720302 Ki = 45 nM T81183 C7PVL8 11730467 IC50 = 2190 nM T81183 CPG15O 11743399 IC50 > 1000 nM T81183 C2J7KO 11751611 Ki = 17.26 nM T81183 CW0UA2 11792453 Ki = 348 nM T81183 CN9M8E 11811722 IC50 = 2830 nM T81183 CN9H3J 11820372 EC50 = 2113 nM T81183 C8EDN0 12088080 Ki = 300 nM T81183 C8RB6W 12088082 Ki > 1000 nM T81183 CRN3S9 13387299 Ki = 9800 nM T81183 CPA2O9 13387301 Ki = 1160 nM T81183 CIDB37 13387304 Ki = 10300 nM T81183 CXS0R8 13387308 Ki = 99000 nM T81183 C1LXY9 13473217 Ki = 6900 nM T81183 C9BQ5D 13473220 Ki = 2000 nM T81183 CLYK03 13538579 Ki = 2250 nM T81183 CES6X1 13538583 Ki = 7400 nM T81183 C36HGR 13538585 Ki = 26000 nM T81183 CV6FD5 13720763 Ki = 1970 nM T81183 CI21BN 14934406 Ki = 17 nM T81183 CAF40B 15181802 IC50 = 8 nM T81183 C2XUE8 15344574 Ki = 36 nM T81183 CEOS76 15523910 Ki = 5915 nM T81183 C6US3O 15711850 Ki > 30000 nM T81183 C5PO3N 15711869 Ki = 1820 nM T81183 CX96HP 18411849 IC50 > 1000 nM T81183 COA7W4 19079030 Ki = 12 nM T81183 CT7XG9 21830793 Ki = 6.75 nM T81183 CYH4J9 22002244 Ki = 0.1 nM T81183 C5SI3U 22464564 Ki = 6780 nM T81183 CJ6WF3 22464606 Ki = 14.8 nM T81183 CA5BY9 22464614 Ki = 8.4 nM T81183 CQB94R 22464634 Ki = 121.1 nM T81183 CAZ23L 22464649 Ki = 13.2 nM T81183 CJCY98 22464720 Ki = 1 nM T81183 CB97XC 22464804 Ki = 4.5 nM T81183 C9MB7K 22464806 Ki = 0.1 nM T81183 C7DXE6 22464831 Ki = 1.7 nM T81183 C76FEA 22464842 Ki = 1.8 nM T81183 C0I2HU 24769156 Ki = 50 nM T81183 C6L7KS 24887518 Ki = 1819.7 nM T81183 C7I9YB 44189144 IC50 = 430 nM T81183 CXR6K7 44212701 Ki > 1000 nM T81183 C8ORL9 44212702 Ki = 2.9 nM T81183 CN71EI 44212703 Ki = 200 nM T81183 C1FRU8 44288600 IC50 > 10000 nM T81183 C7AJ3B 44293793 Ki = 10000 nM T81183 CYUA79 44293794 Ki = 30000 nM T81183 CFDV86 44307552 Ki > 10000 nM T81183 CQRK31 44309145 Ki = 24.4 nM T81183 CHYZ41 44309146 Ki = 91.5 nM T81183 CU2Z3N 44309182 Ki = 2439 nM T81183 CMJV60 44309200 Ki = 5610 nM T81183 C8UR6M 44309202 Ki = 4512 nM T81183 CK26BL 44309367 Ki = 305 nM T81183 C8Y5ZU 44309368 Ki = 610 nM T81183 CHC12P 44309385 Ki = 305 nM T81183 CM02RX 44316058 Ki = 575.44 nM T81183 C9V1IL 44316331 Ki = 389.05 nM T81183 CW16JD 44324737 Ki > 1000 nM T81183 CA84SN 44324765 Ki > 1000 nM T81183 COA3H4 44324800 Ki = 380 nM T81183 CY04JW 44324972 Ki > 1000 nM T81183 C7OW8Y 44336061 Ki = 1118 nM T81183 C4R6LP 44341301 Ki = 23 nM T81183 CD9ZS8 44342270 IC50 = 1150 nM T81183 CJ80OW 44360984 Ki = 28 nM T81183 CS8K1A 44360992 Ki = 18 nM T81183 C3NZ7B 44361021 Ki = 32 nM T81183 CG85AM 44380820 Ki = 730 nM T81183 CT8Y5A 44393007 Ki = 379 nM T81183 CG9S1O 44393045 Ki = 200 nM T81183 CO6EY0 44393113 Ki > 1000 nM T81183 CE03ZW 44393134 Ki = 57 nM T81183 CG5UE1 44393169 Ki = 14 nM T81183 CK85EB 44393193 Ki = 27 nM T81183 CEO2W9 44393372 Ki = 5.8 nM T81183 CXP4Q7 44393393 Ki = 42 nM T81183 C6BZS0 44393403 Ki = 5.9 nM T81183 C86NED 44393411 Ki = 49 nM T81183 C9THO4 44393415 Ki = 1.7 nM T81183 C0E5HY 44400500 Ki = 5.1 nM T81183 CO8EU5 44400519 Ki = 26 nM T81183 CRX12E 44400553 Ki = 35 nM T81183 CIU18E 44400585 Ki = 5.5 nM T81183 CV8K2W 44400594 Ki = 26 nM T81183 C84RNU 44400626 Ki = 73 nM T81183 CY94SF 44400674 Ki = 9.7 nM T81183 CQ4U2P 44403210 Ki = 7.4 nM T81183 CKE6T4 44403213 Ki = 17 nM T81183 CAJX39 44403214 Ki = 12 nM T81183 C61CNS 44403219 Ki = 16 nM T81183 C5AE9L 44403220 Ki = 5.8 nM T81183 CC6XM4 44403224 Ki = 13 nM T81183 C6JB4M 44403225 Ki = 3.9 nM T81183 CGE52H 44403232 Ki = 14 nM T81183 C7W3BP 44405573 Ki = 1.1 nM T81183 CV9IR7 44405574 Ki = 0.5 nM T81183 CFG72V 44405575 Ki = 4 nM T81183 C8WSZ2 44405586 Ki = 0.1 nM T81183 CEJ0C3 44405587 Ki = 0.2 nM T81183 C4DK0U 44405655 Ki = 12.1 nM T81183 C28WCH 44405665 Ki = 18 nM T81183 CS7ZD5 44405666 Ki = 0.2 nM T81183 CIH9J0 44405669 Ki = 0.5 nM T81183 CVZO38 44405677 Ki = 0.5 nM T81183 CMK32Z 44405701 Ki = 26.7 nM T81183 CZK5L6 44405702 Ki = 129.1 nM T81183 CO7G3W 44405725 Ki = 7 nM T81183 CU1VL9 44405726 Ki = 0.2 nM T81183 CO1P3W 44405730 Ki = 1.2 nM T81183 C65PBE 44405930 Ki = 5.47 nM T81183 CBGH16 44405935 Ki = 1.63 nM T81183 CF4S3Y 44405965 Ki = 4.71 nM T81183 CT3Z8U 44405980 Ki = 3.32 nM T81183 CQ7RI8 44405981 Ki = 2.18 nM T81183 C0BI5F 44405985 Ki = 6.28 nM T81183 C1FZE7 44405991 Ki = 1.19 nM T81183 C4NC8M 44405995 Ki = 2.8 nM T81183 CVM1Y5 44406002 Ki = 4.97 nM T81183 C0R5VL 44406003 Ki = 11.71 nM T81183 C90NQJ 44406012 Ki = 4.08 nM T81183 CL5C9T 44406077 Ki = 16.4 nM T81183 C0EXA1 44407083 IC50 > 10000 nM T81183 CG87PW 44409290 Ki > 1000 nM T81183 C2HL9K 44460958 IC50 > 1000 nM T81183 CY8G5Q 44460979 IC50 > 1000 nM T81183 C8T6WQ 46888928 Ki = 2 nM T81183 C18KHC 46888985 Ki = 2 nM T81183 CK40FT 46888986 Ki = 91 nM T81183 CTJ1P2 46889013 Ki = 354 nM T81183 COPQ75 46889014 Ki = 8 nM T81183 CAM45V 46889015 Ki = 46 nM T81183 CZ3FI5 46889016 Ki > 3300 nM T81183 C4B6ZE 46889041 Ki = 1100 nM T81183 C95ZWE 54581386 IC50 > 10000 nM T81183 C2WX4J 54587281 IC50 = 4800 nM T81183 CJZ81X 71293954 Ki = 280 nM T81183 CZ35EN 71294092 Ki = 1.8 nM T81183 CDI84E 71450922 IC50 > 10000 nM T81183 C7W4RH 72734860 Ki = 790 nM T81183 C9T3LW 89638708 Ki = 64 nM T81183 CZDE01 118713090 Ki > 10000 nM T81183 C1KR9C 118713091 Ki = 350 nM T81183 CI5U1R 118713092 Ki = 450 nM T81183 C4S7WD 118713093 Ki = 1.8 nM T81183 CB8Q2E 118713094 Ki = 7.3 nM T81183 C5LFW4 118717221 Ki > 1000 nM T81183 C5OKG2 118727894 Ki = 74.13 nM T81183 CMGB38 118727895 Ki = 89.13 nM T81183 CBHT01 122377930 Ki = 979 nM T81183 CIHZ54 127025242 Ki = 250 nM T81183 CCY7P3 127025243 Ki = 339 nM T81183 CTYP30 127026133 Ki = 742 nM T81183 CX6EI2 127026750 Ki = 1525 nM T81183 C5OU1T 135409492 Ki = 266 nM T81183 C4PM9W 135515431 Ki = 12 nM T81183 CCGZ20 155530937 Ki > 10000 nM T81183 CVBC47 155535120 Ki = 1800 nM T81183 CP9TR0 10324985 Ki = 32.2 nM T81183 D01NOZ 16665072 IC50 = 27000 nM T81183 D02TQC 14928441 Ki = 17000 nM T81183 D04PBA 10015867 Ki > 1000 nM T81183 D05KUM 135446209 Ki = 80 nM T81183 D06HHJ 10490084 Ki = 11000 nM T81183 D09PIF 142067 Ki = 2500 nM T81183 D0A6GK 10489502 Ki = 6000 nM T81183 D0FU5E 10220053 Ki > 1000 nM T81183 D0G2CP 10404144 Ki = 240 nM T81183 D0L6JS 9816048 EC50 = 790 nM T81183 D0N7UE 10198248 Ki = 11000 nM T81183 D0O4BC 11776546 Ki = 5291 nM T81183 D0P5PW 132111 EC50 = 5793 nM T81183 D0S4VR 10655607 Ki = 24000 nM T81183 D0ZC4S 10632290 Ki > 100000 nM T26500 D00KHM 16362 Ki = 2000 nM T26500 D01FGR 3100 Ki = 42657.95 nM T26500 D04USC 774 Ki = 1.6 nM T26500 D08JZS 4992 Ki < 47 nM T26500 D0G8NN 119570 Ki > 10000 nM T26500 D0U5OE 3964 EC50 = 218.78 nM T26500 D0Z1RV 135398737 Ki = 177.83 nM T26500 D01UUD 9948102 Ki > 10000 nM T26500 D02DTQ 24745335 IC50 = 0.65 nM T26500 D07YGH 9976892 Ki > 3162.28 nM T26500 D0M4UZ 24994634 Ki = 12 nM T26500 D0M9RQ 11697697 IC50 > 10000 nM T26500 D0N8QK 24743471 Ki > 10000 nM T26500 D0OW9L 11973780 IC50 > 10000 nM T26500 D02KAF 10103168 EC50 > 0.0001 nM T26500 D05FYA 3035905 Ki = 3.981 nM T26500 D0B4TT 17747460 IC50 = 10000 nM T26500 D0Y2HR 2247 Ki = 7943.28 nM T26500 CMD1L2 5818 Ki = 12.59 nM T26500 C5H9CN 9287 Ki > 10000 nM T26500 CZ1MF7 16106 Ki = 4786.3 nM T26500 CGK70J 16352 Ki = 131.83 nM T26500 CT60VY 32224 Ki < 10000 nM T26500 CXH45A 170389 Ki = 31.62 nM T26500 C2VRP9 182527 EC50 = 8.128 nM T26500 CO5EJ9 206876 Ki = 1000 nM T26500 CWJY10 217674 Ki = 2818.38 nM T26500 C7D4WL 550981 Ki = 2400 nM T26500 CX0ZJ3 565544 EC50 = 549.54 nM T26500 CGY6C5 647957 Ki = 6918.31 nM T26500 C8Q9BF 747187 Ki = 6918.31 nM T26500 CWU5A0 762810 Ki = 6600 nM T26500 C9EGO2 763018 Ki = 6456.54 nM T26500 C61FXJ 767246 Ki = 199.53 nM T26500 CX1Z4F 805994 Ki = 602.56 nM T26500 C9KVI7 832283 Ki = 1071.52 nM T26500 CG53MQ 919019 Ki = 5888.44 nM T26500 CL8OU1 929854 Ki = 5888.44 nM T26500 C0LVU4 933006 Ki = 6309.57 nM T26500 C0RIJ7 1403136 Ki = 1737.8 nM T26500 C1NY7E 1408942 Ki = 199.53 nM T26500 CUVA85 2063135 Ki = 4.7 nM T26500 CUM27P 2306318 Ki = 56 nM T26500 CG0RA3 2971762 Ki = 1479.11 nM T26500 CHS52P 3035746 Ki = 7.8 nM T26500 CAM7I6 3041343 Ki = 489778.82 nM T26500 CRQ6B7 3062060 Ki = 1240 nM T26500 CBE8I7 3076002 Ki = 4073.8 nM T26500 CL3BA9 3201696 IC50 = 20000 nM T26500 CT2A8D 3840250 Ki = 147.91 nM T26500 CUX23E 3934857 IC50 = 37 nM T26500 C1JU8E 3939214 Ki = 7943.28 nM T26500 C9W6SB 3991311 Ki = 269.15 nM T26500 C0OV5H 4060730 Ki = 17 nM T26500 CN3AY7 4242418 Ki = 10000 nM T26500 CJI54B 4242975 Ki = 46 nM T26500 CQ43KY 4563101 Ki = 3162.28 nM T26500 CE1U3D 4687476 Ki = 20400 nM T26500 CQ4JF9 4905344 Ki = 15848.93 nM T26500 C3NM6P 4906599 Ki = 15 nM T26500 C7VR2A 4912179 Ki < 100000 nM T26500 CZ68CO 5159263 Ki = 85 nM T26500 CSEH41 5310982 Ki = 1258.93 nM T26500 C6A9FZ 5477514 Ki = 1480 nM T26500 CSAN19 7015108 Ki = 3500 nM T26500 CJFD94 8070044 Ki = 5754.4 nM T26500 C7IX3U 8070960 Ki = 338.84 nM T26500 C4V5IX 9793791 EC50 = 1096.48 nM T26500 C6HQB2 9793921 Ki = 630.96 nM T26500 CA0K7Q 9839217 Ki = 3 nM T26500 CT5M1L 9851785 Ki > 10000 nM T26500 C0QMJ8 9860842 Ki = 6.31 nM T26500 CW8EZ0 9878733 Ki = 19 nM T26500 C8OTG4 9883231 Ki = 427 nM T26500 CZ34LU 9900313 Ki = 14 nM T26500 CYWQ50 9906447 Ki > 10000 nM T26500 CZ02FE 9923162 Ki = 8 nM T26500 CD50WC 9928073 Ki = 2041.74 nM T26500 CTM0G9 9944571 Ki = 11 nM T26500 CA0B8C 9944610 Ki > 10000 nM T26500 CQ9LU7 9951970 Ki = 1460 nM T26500 CCO8U5 9954017 Ki > 10000 nM T26500 CP9I3U 9964223 Ki = 5128.61 nM T26500 C9X7EB 9965450 Ki = 158.49 nM T26500 CO7GK1 9966927 Ki = 61 nM T26500 C8UE9A 9972181 Ki = 50.12 nM T26500 C3D6KB 9974306 EC50 = 63.1 nM T26500 CN43CY 9990475 Ki = 2511.89 nM T26500 CF7K3Y 9992865 Ki = 19 nM T26500 C58CGU 10017000 Ki = 50.12 nM T26500 CPUJ80 10017821 Ki = 63.1 nM T26500 CG7YZ3 10018335 Ki = 412 nM T26500 CPGA98 10023327 Ki = 12.59 nM T26500 C25DHA 10037650 Ki = 199.53 nM T26500 C32SGR 10041484 Ki = 63.1 nM T26500 CPT7U8 10060212 Ki = 10 nM T26500 CP5L0C 10060213 Ki = 7.943 nM T26500 C12XIY 10063835 Ki = 500 nM T26500 C5Y8BJ 10083188 Ki = 35 nM T26500 CCFP61 10083861 Ki = 528 nM T26500 C3R6NL 10085528 Ki = 63.1 nM T26500 CMKD76 10087533 Ki = 31.62 nM T26500 CT9PI5 10105117 Ki = 25.12 nM T26500 CB0P7C 10106063 EC50 = 77.62 nM T26500 CYQ71B 10107667 Ki = 154 nM T26500 CTZ6D4 10176370 EC50 < 10000 nM T26500 CDM8J7 10197870 Ki = 794.33 nM T26500 CC2MH8 10243990 Ki = 695 nM T26500 C4LA8J 10244243 Ki = 30 nM T26500 C6N1IJ 10261471 EC50 < 10000 nM T26500 C7U0XM 10269628 Ki = 1071.52 nM T26500 CU06TH 10377814 Ki = 316.23 nM T26500 CB2N5K 10399535 Ki = 202 nM T26500 C7GJE9 10419556 Ki = 6309.57 nM T26500 CE8N2K 10429016 Ki = 39.81 nM T26500 C8HVF2 10444761 Ki = 90 nM T26500 CE15WN 10446240 Ki = 63.1 nM T26500 CA76BD 10466840 Ki = 25.12 nM T26500 CA4Z8J 10468601 Ki = 25.12 nM T26500 CI7D9Z 10473209 Ki > 3162.28 nM T26500 CK8NO7 10515050 Ki = 162 nM T26500 C6O1ZI 10515993 Ki = 636 nM T26500 CGW14S 10545988 Ki = 41686.94 nM T26500 C43ACT 10575070 Ki = 17782.79 nM T26500 C6SGD5 10583206 Ki = 2511.89 nM T26500 CX6G7H 10591811 Ki = 27 nM T26500 CU45KX 10656971 Ki = 891.25 nM T26500 CBMH01 10678418 EC50 < 10000 nM T26500 CR8WH9 10678661 Ki = 12589.25 nM T26500 C9O3AL 10688021 Ki = 11 nM T26500 CD7I4S 10702196 Ki = 21877.62 nM T26500 C4DKQ5 10715823 Ki = 779 nM T26500 CWR1T8 10715857 Ki = 118 nM T26500 C56JNC 10760516 Ki = 1548.82 nM T26500 CTG0S1 10773349 Ki = 11748.98 nM T26500 CE8ZO0 10776393 Ki = 118 nM T26500 CF6D2A 10777275 Ki = 426 nM T26500 C36UJO 10782821 Ki = 2691.53 nM T26500 C16RQB 10800875 Ki = 123 nM T26500 C03SWA 10820929 EC50 = 85113.8 nM T26500 CDI46B 10820930 Ki = 12022.64 nM T26500 C45EUI 10860228 Ki = 147 nM T26500 CTC3W5 10879463 Ki = 19952.62 nM T26500 CQS04I 10923241 Ki = 23 nM T26500 CYA27N 10934158 EC50 = 125.89 nM T26500 C2N6AC 10934567 Ki = 31 nM T26500 CX37ZO 10945113 EC50 = 12589.25 nM T26500 C7Y4TW 10957150 Ki = 794.33 nM T26500 C5E7UK 10967174 Ki = 8 nM T26500 CA95TC 10978141 EC50 = 741.31 nM T26500 CF15CY 10986211 EC50 > 0.0001 nM T26500 CSC2B9 10988959 Ki = 15 nM T26500 CKGD62 11013044 Ki = 7000 nM T26500 C1W7ML 11021530 Ki > 10000 nM T26500 C20DCR 11043445 EC50 = 11481.54 nM T26500 C9LE3A 11065080 Ki = 7 nM T26500 CP6E7D 11066922 Ki = 5 nM T26500 CAZ0H8 11086114 EC50 = 7585.78 nM T26500 C6SZ2H 11087453 Ki = 79.43 nM T26500 CO81WF 11094685 EC50 > 0.0001 nM T26500 CWE5L2 11116130 EC50 > 0.0001 nM T26500 CA63ED 11120826 Ki = 32 nM T26500 CUF10O 11126319 EC50 > 0.0001 nM T26500 CU5H7C 11148240 EC50 < 10000 nM T26500 CU9DJ0 11159854 EC50 < 10000 nM T26500 CON91C 11171320 EC50 = 2041.74 nM T26500 C4M9PL 11189343 Ki = 26 nM T26500 CSF2E5 11206058 Ki = 12302.69 nM T26500 CY38JF 11212855 Ki = 93 nM T26500 CIW8G6 11224088 Ki = 1 nM T26500 C6Q8IR 11240759 Ki = 1318.26 nM T26500 CA1XB4 11249610 Ki = 30000 nM T26500 CJ4E3B 11252330 EC50 < 10000 nM T26500 C4XC9T 11258458 Ki = 46 nM T26500 C7G0FN 11258459 Ki = 22 nM T26500 CD3UV9 11275349 EC50 < 10000 nM T26500 CSX09V 11286909 Ki = 1258.93 nM T26500 CLXT61 11293460 Ki = 28 nM T26500 CH05NZ 11340020 Ki = 26 nM T26500 C3HE1G 11344458 Ki = 478.63 nM T26500 CC13FL 11349921 IC50 > 10000 nM T26500 CW3TL6 11408069 Ki = 65 nM T26500 CTP83F 11412714 EC50 < 10000 nM T26500 CG4P9O 11440060 Ki = 240 nM T26500 C40QZP 11451949 Ki = 120 nM T26500 C3B1LH 11469514 Ki = 1000 nM T26500 C7R3SY 11492189 Ki = 630.96 nM T26500 CD4S0X 11499376 Ki = 794.33 nM T26500 CG9Z3H 11499453 Ki = 125.89 nM T26500 CFO2Z5 11499454 Ki = 63.1 nM T26500 CVQR26 11506928 Ki = 50.12 nM T26500 CF45XR 11511026 Ki = 125 nM T26500 CN30CY 11521414 Ki = 100 nM T26500 CL8SY6 11536119 Ki = 50.12 nM T26500 C8GZ1I 11539020 IC50 > 10000 nM T26500 C9UG2V 11544758 Ki > 4000 nM T26500 CY29OV 11546127 Ki = 7780 nM T26500 C0ZBJ6 11554490 Ki = 5.4 nM T26500 CKDY35 11557610 Ki = 39.81 nM T26500 CL3C7W 11564628 Ki = 501.19 nM T26500 C2DKN3 11565330 Ki = 27 nM T26500 CLB3K1 11566111 IC50 = 169 nM T26500 C16AJG 11572015 Ki = 199.53 nM T26500 CGK51J 11572877 Ki = 33 nM T26500 CE0U8J 11581337 IC50 > 10000 nM T26500 C1HJA7 11587279 Ki = 25 nM T26500 C73JSP 11594278 Ki = 7 nM T26500 CN16CW 11600779 Ki = 50.12 nM T26500 CZ79UT 11600780 Ki = 199.53 nM T26500 CN7C5W 11600849 Ki = 158.49 nM T26500 C8E5CJ 11601630 Ki = 40 nM T26500 CIJ8Y1 11609325 Ki = 136 nM T26500 CY4CA7 11615406 Ki = 39.81 nM T26500 C6NZ8Q 11615601 Ki = 158.49 nM T26500 C1N8HD 11615753 Ki = 90 nM T26500 CX2A1I 11622495 Ki = 63.1 nM T26500 CG4HL6 11622672 Ki = 316.23 nM T26500 C6D0VX 11623296 Ki = 49 nM T26500 CW5Z4A 11629829 Ki = 398.11 nM T26500 CP1E8B 11629931 Ki = 501.19 nM T26500 CJ87SH 11630326 Ki = 21 nM T26500 C0G6PN 11632103 IC50 > 10000 nM T26500 C2PGB7 11637064 Ki = 794.33 nM T26500 CPV1Y5 11638468 IC50 = 440 nM T26500 C1R6XC 11672850 Ki = 125.89 nM T26500 C1UGH0 11673377 Ki = 19.95 nM T26500 CL3F6N 11679919 Ki = 316.23 nM T26500 CU5LI1 11679993 Ki = 79.43 nM T26500 CQUT73 11682208 IC50 = 39 nM T26500 C5UDY3 11687917 Ki = 23 nM T26500 CSJ9E7 11688307 Ki = 1960 nM T26500 CU1LP9 11694543 Ki = 100 nM T26500 C7DP1C 11695388 IC50 = 1900 nM T26500 C0SX3K 11701199 Ki = 316.23 nM T26500 C2E8BF 11705395 Ki = 5.2 nM T26500 CA63UW 11708125 Ki = 794.33 nM T26500 CK5ON1 11709443 IC50 = 70 nM T26500 CH51PF 11709905 IC50 = 310 nM T26500 CCS8F5 11724853 Ki = 1412.54 nM T26500 C21NDC 11750684 Ki = 9 nM T26500 C42EXK 11751419 Ki = 250 nM T26500 C9LI8F 11779175 Ki = 447 nM T26500 C7ODJ9 11788475 EC50 < 10000 nM T26500 CMDT64 11804748 EC50 > 0.0001 nM T26500 CYC23D 11819221 EC50 = 741.31 nM T26500 C57IMJ 11821243 Ki = 260 nM T26500 C4JIZ5 11829635 EC50 > 0.0001 nM T26500 COU02Q 11846298 EC50 = 81.28 nM T26500 CE7G4F 11846299 EC50 = 102.33 nM T26500 C0X7FJ 11846300 Ki = 6 nM T26500 CIQ0X2 11846464 EC50 = 14.79 nM T26500 C8J0XO 11846465 Ki = 38.9 nM T26500 CZQX80 11846634 EC50 = 14.79 nM T26500 C0EZ1V 11846635 Ki = 79.43 nM T26500 CR03VI 11846636 EC50 = 20.42 nM T26500 CBOW87 11858011 Ki = 13000 nM T26500 CXLW54 11948707 Ki > 10000 nM T26500 C8JQL7 11957735 IC50 > 10000 nM T26500 CVJ64U 11983344 EC50 = 954.99 nM T26500 CBO10W 12438303 Ki = 2511.89 nM T26500 CNE0A1 12662870 Ki = 251.19 nM T26500 CBZG54 12686452 Ki = 91.2 nM T26500 CTXK62 12686479 Ki = 61.66 nM T26500 CRJ4X2 12741697 Ki = 588.84 nM T26500 C4H1RC 12769844 EC50 = 3630.78 nM T26500 C8OGX6 13153370 Ki < 100000 nM T26500 CPME25 13731320 Ki = 1090 nM T26500 CJ1P9O 14712103 Ki = 630.96 nM T26500 CJ83YW 15984057 Ki = 25118.86 nM T26500 C05CPW 16006947 Ki = 31.2 nM T26500 CNG27H 16061844 Ki = 58 nM T26500 CT6AL1 16061961 EC50 = 20.89 nM T26500 C3ZKG6 16078981 EC50 = 3981.07 nM T26500 CN6V3I 16082820 Ki = 118 nM T26500 C52PUB 16082822 Ki = 143 nM T26500 C5ULI8 16082824 Ki = 115 nM T26500 C9Y8TA 16082826 Ki = 90.4 nM T26500 CV36OS 16082828 Ki = 7.6 nM T26500 CHTO30 16082831 Ki = 37.2 nM T26500 CJ1DV9 16082833 Ki = 127 nM T26500 CFJ53S 16082852 Ki > 1000 nM T26500 CU4KB7 16082854 Ki > 1000 nM T26500 CW9SA4 16082856 Ki = 130 nM T26500 CRP4X3 16082858 Ki = 177 nM T26500 CT2NF0 16082860 Ki = 103 nM T26500 CIP39S 16082862 Ki > 1000 nM T26500 CT9B1U 16082864 Ki > 1000 nM T26500 C3YF6A 16082866 Ki > 1000 nM T26500 CYEG41 16202258 Ki = 0.034 nM T26500 CMF2I1 16656869 IC50 = 1600 nM T26500 C03TDU 16656870 IC50 = 95 nM T26500 C3T2ZK 16656871 IC50 = 285 nM T26500 CSZ62L 16656872 IC50 = 33 nM T26500 CY4LM7 16656874 IC50 = 87 nM T26500 C08XJA 16718567 Ki = 0.4 nM T26500 C9RK0S 20299674 Ki = 10 nM T26500 C1JN0B 21029584 Ki = 328 nM T26500 C5JCZ6 21193534 Ki = 25 nM T26500 C54PIH 21638785 Ki = 12.59 nM T26500 CDS1G7 21842421 Ki = 1099 nM T26500 CHI0K9 21896704 Ki = 214 nM T26500 C82PTR 22660598 Ki = 2511.89 nM T26500 C6NY1Z 22660616 Ki = 25.12 nM T26500 C3BP7D 23151209 IC50 > 10000 nM T26500 CV6A0G 23649429 Ki = 57.54 nM T26500 C0KS2V 23650959 Ki = 5 nM T26500 CA2M0O 23653543 Ki = 0.1 nM T26500 CTZL46 24278976 Ki = 229.09 nM T26500 CTM7A2 24729202 EC50 < 10000 nM T26500 C0JS9D 24737947 Ki = 3.4 nM T26500 CIG74O 24737949 Ki = 2 nM T26500 CO1UT8 24737950 Ki = 0.7 nM T26500 CSM09I 24737952 Ki = 11 nM T26500 C5N4DE 24737954 Ki = 10 nM T26500 CZD42M 24738103 Ki = 20 nM T26500 CLVB35 24738269 Ki = 2.4 nM T26500 CM0R5W 24739219 Ki = 19 nM T26500 CZO1Q2 24745337 Ki = 4 nM T26500 CZ6T4O 24745506 Ki = 1.5 nM T26500 C0Z5WO 24745507 Ki = 13 nM T26500 CAVZ24 24759518 Ki = 104.71 nM T26500 CQ5S2G 24759622 Ki = 7585.78 nM T26500 C21BRL 24759624 Ki = 26.3 nM T26500 CMC47K 24764570 Ki = 630.96 nM T26500 CLDQ41 24797248 EC50 = 43.65 nM T26500 C5D1MS 24797598 Ki = 1 nM T26500 C4ONS7 24797604 Ki = 1.4 nM T26500 C24PAD 24797956 Ki = 5.5 nM T26500 C5Z1AB 24798144 Ki = 1 nM T26500 CT9R2H 24798232 Ki = 1.8 nM T26500 CJM86D 24798596 EC50 = 37.15 nM T26500 CLB5M8 24825514 Ki = 5.623 nM T26500 C8DQR0 24825515 Ki = 5.623 nM T26500 CIM1V9 24825522 Ki = 8.318 nM T26500 CN6JR4 24825727 Ki = 1.1 nM T26500 C0I1TN 24825791 Ki = 5.7 nM T26500 C0IJC6 24825794 Ki = 9.1 nM T26500 CTY73E 24825796 Ki = 137 nM T26500 C8SGX6 24825897 Ki = 29 nM T26500 CGT20B 24825995 Ki = 65 nM T26500 COL1H0 24825996 Ki = 2.1 nM T26500 CDR1G5 24825998 Ki = 1 nM T26500 CFZ4K1 24825999 Ki > 10000 nM T26500 C0R3PQ 24826000 Ki = 125 nM T26500 CK98HD 24826080 Ki = 440 nM T26500 C1E3UF 24826081 Ki = 43 nM T26500 CPQ03L 24826082 Ki = 25 nM T26500 C10WGD 24826083 Ki = 149 nM T26500 CQWC96 24826162 Ki = 5.2 nM T26500 CY7JB3 24826163 Ki = 33 nM T26500 C1HMA5 24826165 Ki = 18 nM T26500 C1JNC8 24826167 Ki = 76 nM T26500 CMWQ23 24826168 Ki = 10 nM T26500 CXGP32 24826169 Ki = 0.3 nM T26500 C8RQW4 24826265 Ki = 19 nM T26500 CYI9M6 24826268 Ki = 75 nM T26500 CV6X9L 24826354 Ki = 31 nM T26500 C4HN5A 24826358 Ki = 3.6 nM T26500 CUT52P 24826437 Ki = 4.7 nM T26500 C1JLU9 24826438 Ki > 10000 nM T26500 C0VS1Y 24826439 Ki = 47 nM T26500 C12YVI 24826440 Ki > 10000 nM T26500 CJ5VN7 24826441 Ki = 30 nM T26500 C06XVY 24826442 Ki = 12 nM T26500 C6HO2R 24826443 Ki = 121 nM T26500 C8GH0O 24826518 Ki = 50 nM T26500 C6B0SH 24826519 Ki > 10000 nM T26500 CA2R7Y 24826522 Ki = 10 nM T26500 CV4AF0 24826598 Ki = 363 nM T26500 CB03ME 24826679 Ki = 74 nM T26500 C2U1FY 24826680 Ki = 40 nM T26500 CW6V8K 24826681 Ki = 1049 nM T26500 CX6V2W 24826682 Ki > 10000 nM T26500 C1BF5A 24826766 Ki = 0.9 nM T26500 CZQ7U8 24827129 Ki = 8 nM T26500 CG7KM8 24853527 Ki = 1548.82 nM T26500 CMV45T 24853528 Ki = 3981.07 nM T26500 CUF5V6 24853529 Ki = 363.08 nM T26500 C53RSE 24853592 Ki = 2951.21 nM T26500 C8QB6R 24853593 Ki = 4365.16 nM T26500 CDP08X 24853594 Ki = 1380.38 nM T26500 CZL4S6 24853595 Ki = 269.15 nM T26500 CA9RT3 24853596 Ki = 2344.23 nM T26500 CK8YE0 24853597 Ki = 575.44 nM T26500 C8Y5JD 24853598 Ki = 2344.23 nM T26500 CL45DZ 24853662 Ki = 13182.57 nM T26500 C4I8QS 24853663 Ki = 229.09 nM T26500 CF1BT7 24853664 Ki = 1174.9 nM T26500 CVE0S8 24853666 Ki = 977.24 nM T26500 C4QHJ1 24854583 Ki = 10232.93 nM T26500 CF0WA5 24854634 Ki = 3981.07 nM T26500 C7QCD3 24854635 Ki = 63.1 nM T26500 CRQ13Y 24854636 Ki = 2511.89 nM T26500 CRU2Y0 24854637 Ki = 323.59 nM T26500 C0YUJ2 24854638 Ki = 295.12 nM T26500 C5BH7U 24854639 Ki = 478.63 nM T26500 CK1OB2 24854640 Ki = 467.74 nM T26500 CRF78N 24854702 Ki = 2951.21 nM T26500 CKZU49 24854703 Ki = 707.95 nM T26500 C3S4BL 24854704 Ki = 2290.87 nM T26500 COZ2N0 24854705 Ki = 1288.25 nM T26500 CX1V6F 24854706 Ki = 1698.24 nM T26500 C1V5FE 24854707 Ki = 1584.89 nM T26500 C0RWT3 24854708 Ki = 2187.76 nM T26500 CZPW63 24936097 Ki > 1000 nM T26500 CQ52SD 24936098 Ki > 1000 nM T26500 CE9R4B 24948752 Ki = 1.1 nM T26500 CWA0R4 24978528 Ki = 15.85 nM T26500 C4ZYR1 24992077 Ki = 1.5 nM T26500 C07HDB 24992735 Ki = 43 nM T26500 C9PVA7 24994542 Ki = 1.1 nM T26500 CERP91 24994630 Ki = 257 nM T26500 CU94JC 24994635 Ki = 12 nM T26500 CY51IA 24994636 Ki = 30 nM T26500 C0QW7C 24994945 Ki = 77 nM T26500 C62TBC 24994950 Ki = 357 nM T26500 CGRH31 24996854 Ki = 11.2 nM T26500 C2G1JK 25053351 Ki > 10000 nM T26500 CLQ5Z0 25071004 Ki = 3.467 nM T26500 CVP3S9 25071319 Ki = 70.79 nM T26500 CPR94U 25071940 Ki = 52.48 nM T26500 C51OJR 25099115 IC50 > 10000 nM T26500 CYD90E 25101945 Ki = 10.96 nM T26500 C7NJ1B 25109291 Ki = 5.754 nM T26500 CHP82T 25112105 Ki = 2 nM T26500 CML6G5 25128822 Ki = 15.49 nM T26500 C6DC9I 25128823 Ki = 12.88 nM T26500 C6WA8X 25128824 Ki = 5.1 nM T26500 C3SXH2 25128831 EC50 = 11481.54 nM T26500 CP3QM7 25128833 Ki = 31 nM T26500 C7QMJ4 25129169 Ki = 39.8 nM T26500 CAGM54 25129523 Ki = 5.012 nM T26500 C94BRW 25129525 Ki = 15.85 nM T26500 CI8V3B 25129527 Ki = 1.995 nM T26500 C4ZLI1 25130230 EC50 = 2511.89 nM T26500 C6FWM1 25130231 EC50 = 177.83 nM T26500 CEJ0O4 25130236 EC50 = 4897.79 nM T26500 C7JU1L 25130576 Ki = 41.69 nM T26500 CPU26L 25130581 EC50 = 1202.26 nM T26500 CC9ML0 25130909 EC50 = 33.88 nM T26500 CX0JH8 25130912 Ki = 6 nM T26500 C8LMG6 25130914 EC50 = 12.59 nM T26500 CML37J 25131556 EC50 = 26.92 nM T26500 CAUP56 25131559 EC50 = 16.22 nM T26500 CA9B8N 25131561 EC50 = 3890.45 nM T26500 C1PA7L 25133970 Ki = 1081 nM T26500 CR7QT9 25133972 EC50 = 2344.23 nM T26500 C6HD3B 25147771 Ki = 26.92 nM T26500 C1RU5I 25147772 Ki = 7.586 nM T26500 C8D7HZ 25149335 EC50 = 15.14 nM T26500 CQ7N3X 25149521 EC50 = 7.943 nM T26500 C92NXM 25149613 EC50 = 66.3 nM T26500 C4GC8J 25149708 EC50 = 6.3 nM T26500 C6NAC0 25149712 EC50 = 15.85 nM T26500 C26OMF 25178130 Ki = 8511.38 nM T26500 C0AG1S 25178131 Ki = 239.88 nM T26500 CXWJ98 25178132 Ki = 758.58 nM T26500 C9R3VG 25178339 Ki = 588.84 nM T26500 CQE0B9 25178340 Ki = 954.99 nM T26500 CXF28Y 25178341 Ki = 562.34 nM T26500 C18FSV 25178342 Ki = 104.71 nM T26500 CBPJ78 25178343 Ki = 128.82 nM T26500 CLVH57 25178344 Ki = 436.52 nM T26500 C0BHA6 25178345 Ki = 89.13 nM T26500 C8S1HC 25178551 Ki = 223.87 nM T26500 CO0R5Y 25178552 Ki = 60.26 nM T26500 C5TMN4 25178553 Ki = 38.9 nM T26500 CSE76V 25178554 Ki = 371.54 nM T26500 C39JAH 25178555 Ki = 107.15 nM T26500 C1TJH2 25178556 Ki = 269.15 nM T26500 C5FMI4 25178558 Ki > 1000 nM T26500 C19NAF 25178750 Ki > 1000 nM T26500 C05QSD 25178752 Ki > 1000 nM T26500 CT01VH 25178755 Ki = 154.88 nM T26500 C2HE6Q 25178756 Ki > 1000 nM T26500 CYR8K6 25178758 Ki > 1000 nM T26500 CP7I5E 25178759 Ki > 1000 nM T26500 CF9UI4 25178760 Ki > 1000 nM T26500 CJ5EH8 25178933 Ki = 257.04 nM T26500 C7C9LH 25178936 Ki = 616.6 nM T26500 C59YLX 25178937 Ki = 70.79 nM T26500 C6N8HW 25178938 Ki = 630.96 nM T26500 CTD19J 25178939 Ki = 363.08 nM T26500 CJS1H4 25179122 Ki = 186.21 nM T26500 CEO06R 25179123 Ki = 891.25 nM T26500 CV57PI 25179124 Ki = 186.21 nM T26500 C0VM8R 25179125 Ki = 35.48 nM T26500 C27QSA 25179126 Ki = 134.9 nM T26500 CLWJ25 25179127 Ki = 33.88 nM T26500 CX1J7W 25179297 Ki = 104.71 nM T26500 C5N8MJ 25179299 Ki > 1000 nM T26500 C2Y3JU 25179300 Ki > 1000 nM T26500 CX38LG 25179302 Ki > 1000 nM T26500 C3DJ8W 25179303 Ki = 141.25 nM T26500 CX2R6Z 25179304 Ki > 1000 nM T26500 CYW92S 25179305 Ki > 1000 nM T26500 CE0N1C 25179493 Ki > 1000 nM T26500 CZ4KX1 25217643 Ki = 10 nM T26500 CUK5E6 25218146 Ki = 21 nM T26500 C73KWR 29136870 Ki = 2900 nM T26500 CDZ54N 35665437 Ki < 100000 nM T26500 CUN63T 39732699 Ki = 100 nM T26500 CI7RK5 42624148 Ki = 28 nM T26500 CN7KY1 42624149 Ki = 21 nM T26500 CXOH20 42624150 Ki = 8 nM T26500 CMKQ63 42625221 EC50 = 7.079 nM T26500 CIJ52Y 42625222 EC50 = 28.18 nM T26500 CR7LN9 42625223 EC50 = 151.36 nM T26500 C8G7QX 42625303 EC50 = 3.02 nM T26500 C75WJN 42625304 EC50 = 3.715 nM T26500 C0BW6J 42625384 EC50 = 4.898 nM T26500 CID4J1 42625386 EC50 = 2.57 nM T26500 C5YR2D 42626109 EC50 = 19.05 nM T26500 CI34UC 42626111 EC50 = 33.11 nM T26500 CQN2L0 42641407 Ki = 151.36 nM T26500 C46ULX 43398194 Ki = 398.11 nM T26500 CFL6W8 44126357 Ki = 320 nM T26500 C1VUR5 44129056 Ki = 5.37 nM T26500 CEH53X 44129130 Ki = 4 nM T26500 CH67CD 44129131 Ki = 7.586 nM T26500 C3N6LO 44129132 Ki = 12.59 nM T26500 C3GL8J 44129133 Ki = 4.266 nM T26500 CNS28O 44129134 Ki = 4.467 nM T26500 C9X8OD 44129135 Ki = 9.333 nM T26500 C2RCJ5 44129209 Ki = 70.79 nM T26500 COK43R 44129210 Ki = 33.11 nM T26500 C2EYU3 44129211 Ki = 26.92 nM T26500 CMBN73 44129212 Ki = 8.128 nM T26500 CQ52HF 44129213 Ki = 19.05 nM T26500 C1WUP6 44129214 Ki = 15.49 nM T26500 C6BH3A 44129282 Ki = 11.22 nM T26500 C4HD5M 44129283 Ki = 309.03 nM T26500 CYL93A 44187557 Ki = 1.585 nM T26500 C6P7EH 44211094 EC50 < 10000 nM T26500 CL2IE8 44231618 Ki = 1.514 nM T26500 CP5MX1 44231735 Ki = 1.995 nM T26500 C8P2LE 44250288 IC50 > 10000 nM T26500 C5YFB9 44252324 IC50 > 10000 nM T26500 CVQ13I 44275465 Ki = 32 nM T26500 CE20CZ 44275807 Ki = 10000 nM T26500 CS0E2H 44367567 EC50 = 416.87 nM T26500 CS2J8O 44367568 EC50 = 1023.29 nM T26500 C8KPD7 44395263 Ki = 25118.86 nM T26500 CSV36Q 44395290 Ki = 25118.86 nM T26500 CY51NG 44395308 Ki = 63.1 nM T26500 CUW8B3 44395314 Ki = 5011.87 nM T26500 CHU6B8 44395335 Ki = 1000 nM T26500 CIK6G0 44395336 Ki = 25118.86 nM T26500 CX2JT9 44395361 Ki = 19952.62 nM T26500 C9QSE7 44395364 Ki = 199.53 nM T26500 CGVU87 44395388 Ki < 100000 nM T26500 C4E8JC 44395389 Ki < 100000 nM T26500 C9X2SV 44414433 Ki = 6456.54 nM T26500 CC51VO 44414495 Ki = 13803.84 nM T26500 CH7D4C 44414498 Ki = 6456.54 nM T26500 C0WBD5 44450401 Ki = 1479.11 nM T26500 C5J4MD 44450438 Ki = 7413.1 nM T26500 C0VBW1 44450493 Ki = 11.75 nM T26500 CB74AR 44462956 Ki = 7.079 nM T26500 CQ0WM7 44469273 IC50 > 5000 nM T26500 CK10AW 44478385 EC50 = 33.88 nM T26500 CJ27OY 44480707 EC50 = 1288.25 nM T26500 CR6G8Q 44480708 EC50 = 1096.48 nM T26500 C4ELF5 44480958 EC50 = 2570.4 nM T26500 C7GMD8 44480959 EC50 = 169.82 nM T26500 CM4GV5 44480960 EC50 = 331.13 nM T26500 CO5S2C 44481486 EC50 > 10000 nM T26500 C3SJ9D 44481489 EC50 = 758.58 nM T26500 C53ROK 44481761 EC50 = 151.36 nM T26500 C2LH9Y 44482028 EC50 = 575.44 nM T26500 CPF2E9 44482029 EC50 = 1202.26 nM T26500 CSK27P 44482030 EC50 = 141.25 nM T26500 CG7W2C 44482031 EC50 = 707.95 nM T26500 C5K8QN 44482032 EC50 = 120.23 nM T26500 CQZ64I 44482298 EC50 > 10000 nM T26500 C0PR2N 44546966 Ki = 51 nM T26500 CFO68H 44547126 Ki = 96 nM T26500 C3SHB9 44547127 Ki = 19 nM T26500 CV6E5Y 44547268 Ki = 2 nM T26500 C47FYK 44547564 Ki = 16 nM T26500 C28QZX 44547567 Ki = 33 nM T26500 CVHT72 44547568 Ki = 109 nM T26500 CA36FX 44563707 Ki = 269.15 nM T26500 COF8M1 44576985 Ki = 897 nM T26500 C9DVO6 44595856 Ki = 6.31 nM T26500 C8JQ4C 44609412 Ki = 7.943 nM T26500 CEW8Y5 44628629 Ki = 21 nM T26500 CIL8V6 44628631 Ki = 138 nM T26500 CYXD79 45257131 EC50 = 8.511 nM T26500 C07WHQ 45257132 EC50 = 1.122 nM T26500 CY25IH 45257133 EC50 = 6.026 nM T26500 CM14OG 45257134 EC50 = 269.15 nM T26500 C5ND1K 45263439 Ki = 31.62 nM T26500 CQ5NW7 45263442 Ki = 7943.28 nM T26500 CK9C2R 45263443 Ki = 3162.28 nM T26500 C72OTL 45263460 Ki = 3981.07 nM T26500 CB0DY2 45265852 Ki = 398.11 nM T26500 CQH4L3 45267230 Ki = 10 nM T26500 C3X7CM 45267233 Ki = 12.59 nM T26500 C46QKW 45267237 Ki = 100 nM T26500 CWL5Y3 45268093 Ki = 10 nM T26500 CEJ07N 45268095 Ki = 25.12 nM T26500 CUG4V7 45268970 Ki = 158.49 nM T26500 CF36SE 45269820 EC50 = 6.31 nM T26500 C5YUW8 45270644 Ki = 25.12 nM T26500 C24QGO 45271464 Ki = 25.12 nM T26500 CC85BP 45271470 Ki = 25.12 nM T26500 CQFK46 45379805 Ki = 17.78 nM T26500 CAY1O3 45379807 Ki = 223.87 nM T26500 CTVH35 45379808 Ki = 489.78 nM T26500 C5E6OH 45379921 Ki = 50.12 nM T26500 CW15UK 45379922 Ki = 5.754 nM T26500 C3QU2C 45487384 IC50 > 5000 nM T26500 CC04ZF 46228069 Ki = 8100 nM T26500 C09ILM 46228070 Ki = 35000 nM T26500 C7RX0E 46228071 Ki = 207 nM T26500 CCL6R1 46228076 Ki = 3400 nM T26500 CP58OH 46228082 Ki = 2200 nM T26500 CXG9U1 46228083 Ki = 716 nM T26500 C8SW9C 46228087 Ki = 376600 nM T26500 C02QAD 46228092 Ki = 2500 nM T26500 CXDY71 46228100 Ki = 13700 nM T26500 C36VJG 46228101 EC50 = 31.62 nM T26500 C9OEB4 46228113 Ki = 542 nM T26500 C08QZB 46228114 EC50 = 102.33 nM T26500 C4Q8ZJ 46228125 EC50 = 56.23 nM T26500 C19VQX 46228126 Ki = 1200 nM T26500 CWO1R9 46228132 EC50 = 104.71 nM T26500 CVRQ29 46228133 EC50 = 199.53 nM T26500 C6YI0N 46228143 EC50 = 478.63 nM T26500 C4N7MG 46228158 Ki = 341 nM T26500 CT4HX9 46228994 Ki = 10 nM T26500 CU15OL 46235428 Ki = 0.21 nM T26500 CN75IJ 46830167 EC50 = 2.63 nM T26500 CPDQ25 46881855 Ki = 48.98 nM T26500 CK8LF2 46884945 IC50 = 10000 nM T26500 CG63KP 46884996 IC50 = 236 nM T26500 CXSO17 46884997 IC50 = 21000 nM T26500 C7H1YU 46884998 IC50 = 126 nM T26500 CD7B5Y 46885127 IC50 > 10000 nM T26500 CLF31Q 46885128 IC50 = 1400 nM T26500 CJ0Q9Z 46885129 IC50 = 1400 nM T26500 CD62KF 46885130 IC50 > 10000 nM T26500 CG8JD1 46885131 IC50 > 10000 nM T26500 C9LI0J 46885177 IC50 = 86 nM T26500 CIN2X7 46885178 IC50 = 30 nM T26500 C0RM5L 46885179 IC50 > 10000 nM T26500 CG5W3O 46885180 IC50 > 30000 nM T26500 C8SQB9 46885181 IC50 = 6200 nM T26500 CAYE16 46885182 IC50 > 30000 nM T26500 CM4BA7 46885239 IC50 = 171 nM T26500 CH2QO5 46885240 IC50 > 30000 nM T26500 CQVF63 46885241 IC50 = 14200 nM T26500 C1S9GV 46885296 IC50 > 10000 nM T26500 CET5L8 46885297 IC50 = 1000 nM T26500 CJX6L2 46885298 IC50 = 90 nM T26500 CB29TI 46887041 EC50 = 22.91 nM T26500 C9P3CV 46887042 EC50 = 8.318 nM T26500 C12SYH 46887043 EC50 = 4.571 nM T26500 CQJ8W2 46887076 EC50 > 10000 nM T26500 CAG89L 46887077 EC50 > 10000 nM T26500 COK81L 46887078 EC50 > 10000 nM T26500 CB09SD 46887079 EC50 = 6025.6 nM T26500 CK0S2U 46887080 EC50 > 10000 nM T26500 CLPJ52 46887115 EC50 = 1380.38 nM T26500 C8RL6E 46890019 Ki = 77 nM T26500 C26JVO 46890020 Ki = 150 nM T26500 CPH7R6 46890021 Ki = 1756 nM T26500 C4MZ5E 46890022 EC50 = 6.9 nM T26500 CKY32V 46890071 Ki = 557 nM T26500 C1I3BG 46890072 EC50 = 3.3 nM T26500 CL14XI 46890073 Ki > 10000 nM T26500 CXKH26 46890074 Ki = 152 nM T26500 CZM95N 46890120 Ki = 228 nM T26500 CA1WZ2 46890121 Ki > 10000 nM T26500 CW10LT 46890122 Ki = 133 nM T26500 COR71G 46890166 Ki = 3.3 nM T26500 CN1O2I 46890167 Ki = 609 nM T26500 C7O1DR 46890200 Ki = 5000 nM T26500 C3X0HK 46890545 Ki = 32 nM T26500 CO39UY 46890546 Ki = 80 nM T26500 CUQJ21 46890547 Ki = 20 nM T26500 CLZK09 46890548 Ki = 84 nM T26500 C57SMC 46890549 Ki = 72 nM T26500 CIZ95Y 46890589 Ki = 2000 nM T26500 CYI3B2 46890590 Ki = 42 nM T26500 C5JR8C 46890591 Ki = 1000 nM T26500 C8FR9E 46890592 Ki = 14 nM T26500 C7TK0P 46890626 Ki = 691 nM T26500 CSO98E 46890627 Ki = 26 nM T26500 CHAY62 46890628 Ki > 10000 nM T26500 CT0R2K 46890629 Ki > 10000 nM T26500 CNPM18 46890674 Ki > 10000 nM T26500 CD7XP9 46890675 Ki = 232 nM T26500 C9DRX2 46890676 Ki = 971 nM T26500 CP0U2A 46890677 Ki = 89 nM T26500 CDV30W 46912441 Ki = 216 nM T26500 CAQ0E9 46912442 Ki = 3100 nM T26500 C6F2MP 46929551 Ki = 840 nM T26500 CT3UX6 46929553 Ki = 360 nM T26500 CZJ2G8 46929554 Ki = 17 nM T26500 C40EGB 46929647 Ki = 1300 nM T26500 CB95RA 46929648 Ki = 310 nM T26500 CN39XY 49818718 Ki = 24 nM T26500 CMD1V2 49841607 Ki = 91 nM T26500 CH13RK 49841608 Ki = 17 nM T26500 C08MLJ 49841609 Ki = 111 nM T26500 CN9SO5 49841610 Ki = 19 nM T26500 C63YRM 49841611 Ki = 90 nM T26500 CM6YL4 49841612 Ki = 29 nM T26500 CKNW10 49841718 Ki = 55 nM T26500 CG97QN 49841719 Ki = 4 nM T26500 CR52VK 49841720 Ki = 32 nM T26500 CVQ18H 49841721 Ki = 221 nM T26500 CWI59B 49841722 Ki = 2333 nM T26500 CEC6Y1 49841723 Ki = 945 nM T26500 CZ3T1W 49841845 Ki = 5 nM T26500 C3SBE0 49841846 Ki = 3 nM T26500 CM0TG4 49841962 Ki = 109 nM T26500 C3KF6B 49865668 Ki = 51 nM T26500 C2RY0J 50878551 Ki > 10000 nM T26500 C1W6TV 50898777 Ki > 10000 nM T26500 CXMZ73 50898778 Ki > 10000 nM T26500 CE4KP1 51050257 Ki > 10000 nM T26500 C1IL7V 51354008 Ki = 1148.15 nM T26500 CCX8V5 51354009 Ki = 181.97 nM T26500 CC0QD5 51354010 Ki = 912.01 nM T26500 C2RY8V 51354296 Ki = 1819.7 nM T26500 CLFW43 51354297 Ki = 15135.61 nM T26500 CEL4X0 51354298 Ki = 100 nM T26500 C3OT2L 51354299 Ki = 67.61 nM T26500 CYHG32 51354300 EC50 = 1 nM T26500 CDY7Q9 51354301 EC50 = 125.89 nM T26500 CQ1S6T 51354302 Ki = 275.42 nM T26500 C1U6YS 51354303 Ki = 89.13 nM T26500 CX8AQ3 51354304 Ki = 141.25 nM T26500 CSHG49 51354581 Ki = 457.09 nM T26500 C8GQM0 51354582 Ki = 21.38 nM T26500 CL0QJ4 51354583 Ki = 54.95 nM T26500 C9S6YJ 51354584 Ki = 7.943 nM T26500 C3UBQ6 51354585 Ki = 588.84 nM T26500 CFG8J0 51354586 Ki = 1148.15 nM T26500 C5OC9L 51354587 Ki = 21877.62 nM T26500 C08AOI 51354588 Ki = 4786.3 nM T26500 CI9YD2 51354870 Ki = 20892.96 nM T26500 CHN6Q5 51354871 Ki = 11220.18 nM T26500 C0V7HN 51354872 Ki = 38904.51 nM T26500 C54XUL 51354873 Ki = 446.68 nM T26500 C2DHY5 51354874 Ki = 446.68 nM T26500 CK5N0S 51354875 Ki = 79.43 nM T26500 CB54WT 51354877 Ki = 380.19 nM T26500 CE2R6U 51355156 Ki = 251.19 nM T26500 C4E9MQ 51355443 Ki = 588.84 nM T26500 CTDU94 52128564 Ki = 251.19 nM T26500 CC2Q0P 52952957 Ki = 7079.46 nM T26500 C5D7WN 53233801 Ki = 15 nM T26500 CBR65J 53233802 Ki = 10 nM T26500 C7RY0U 53233803 Ki = 28 nM T26500 CRDB36 53233804 Ki = 3 nM T26500 C7EPV6 53233805 Ki = 2 nM T26500 C51HOU 53233904 Ki = 100 nM T26500 C4Y0DA 53257796 Ki = 2.4 nM T26500 CJ31IK 53258370 Ki = 21 nM T26500 C1L7WJ 53321919 Ki = 7.943 nM T26500 CA2U6E 53378711 Ki = 9.4 nM T26500 C8JQ0L 53378928 Ki = 16 nM T26500 C1TNU0 53378933 Ki = 100 nM T26500 CT19XH 53476465 Ki = 3.4 nM T26500 C7MG8L 54580746 Ki = 8 nM T26500 CF90XI 54580885 Ki = 0.9 nM T26500 CTL98P 54581937 Ki = 189 nM T26500 CRZQ23 54581938 Ki = 77 nM T26500 CY42ZV 54581939 Ki = 853 nM T26500 CC8G5A 54581940 Ki = 1 nM T26500 C69ORU 54581941 Ki = 40 nM T26500 CG3KU6 54582865 Ki = 6 nM T26500 C87AUN 54582866 Ki = 1076 nM T26500 C0T5KW 54582867 Ki = 24 nM T26500 CHM1X4 54583872 Ki = 69 nM T26500 C35ICE 54583873 Ki = 3 nM T26500 C8E0MB 54583874 Ki = 132 nM T26500 CM01JW 54583875 Ki = 36 nM T26500 CZ34PR 54584374 Ki = 3801.89 nM T26500 CFDA28 54584378 Ki = 13182.57 nM T26500 C7RT1W 54584824 Ki = 3 nM T26500 C8EIU7 54584825 Ki = 6 nM T26500 C58CJV 54584826 Ki = 127 nM T26500 C41PQB 54584827 Ki = 83 nM T26500 C42ICP 54585776 Ki = 255 nM T26500 CG5BD8 54585777 Ki = 50 nM T26500 C4BE6K 54585778 Ki = 1155 nM T26500 CC5JW1 54585779 Ki = 140 nM T26500 C4CW2L 54585780 Ki = 3 nM T26500 CE91SF 54585781 Ki = 2 nM T26500 C7DZ0P 54586762 Ki = 148 nM T26500 C8AQE3 54586763 Ki = 0.3 nM T26500 C48UWH 54586764 Ki = 51 nM T26500 CBD1E2 54586765 Ki = 44 nM T26500 C96ZCR 54587786 Ki = 29 nM T26500 C39JDB 54587787 Ki = 0.2 nM T26500 C0DUZ1 54587788 Ki = 0.04 nM T26500 CFI18A 54587789 Ki = 25 nM T26500 CQ7R0C 54587790 Ki = 9 nM T26500 CLBQ29 54587791 Ki = 162 nM T26500 C6ULC1 54587792 Ki = 64 nM T26500 C5OBC3 54753437 Ki = 9 nM T26500 CB72FX 54754351 Ki = 37 nM T26500 CPS5V6 54764158 Ki > 10000 nM T26500 C9OUQ6 54765288 IC50 > 10000 nM T26500 CWL5O1 55251397 Ki = 277 nM T26500 CHJ2C7 56593499 EC50 = 110 nM T26500 CU01AZ 56659113 Ki = 288.4 nM T26500 C53IST 56672434 Ki = 794.33 nM T26500 CG5U0K 56682943 Ki = 323.59 nM T26500 CY92VU 56835087 Ki > 10000 nM T26500 C0JMA7 56835088 Ki > 10000 nM T26500 C4E6HV 56835171 Ki = 7 nM T26500 CND5M6 56849569 Ki = 125.89 nM T26500 C6Y4GM 56849571 Ki = 134.9 nM T26500 C7YVT9 56851441 Ki = 42.66 nM T26500 CN0P6H 56851443 Ki = 75.86 nM T26500 C7VE0O 56851445 Ki = 16.22 nM T26500 CBW34E 56851447 Ki = 147.91 nM T26500 C6XG8Z 56851602 Ki = 89.13 nM T26500 CQ51VT 56851604 Ki = 229.09 nM T26500 CGO4X5 56851606 Ki = 380.19 nM T26500 C4QHS9 56851608 Ki = 31.62 nM T26500 CQOE56 56851610 Ki = 29.51 nM T26500 CCO25Y 56851612 Ki = 89.13 nM T26500 CS5VP4 56950378 Ki = 52 nM T26500 C7B8RI 56954318 EC50 = 79.43 nM T26500 C7G3TI 56954320 EC50 = 41.69 nM T26500 CKG35O 56954322 EC50 = 8.511 nM T26500 CI7XO6 56954425 EC50 = 338.84 nM T26500 C2W9CZ 56954427 EC50 > 1000 nM T26500 CIQH95 56954515 EC50 = 8.511 nM T26500 C1TC7Q 56963799 Ki > 10000 nM T26500 CO9RV4 57328003 Ki >= 31622.78 nM T26500 CS2PJ1 57328076 Ki >= 31622.78 nM T26500 CYHP54 57328077 Ki >= 31622.78 nM T26500 C9TOC0 57328078 Ki >= 31622.78 nM T26500 CW1YS8 57328079 Ki >= 31622.78 nM T26500 C5J8EQ 57328080 Ki >= 31622.78 nM T26500 C4HUF2 57328081 Ki >= 31622.78 nM T26500 C50CFD 57328141 Ki >= 31622.78 nM T26500 CKB8T1 57328142 Ki >= 31622.78 nM T26500 CT92DL 57328143 Ki >= 31622.78 nM T26500 CEO74T 57328144 Ki >= 31622.78 nM T26500 CD5GS3 57328145 Ki >= 31622.78 nM T26500 C25AFJ 57328146 Ki >= 31622.78 nM T26500 CG80ZN 57328209 Ki >= 31622.78 nM T26500 CT2F3I 57328210 Ki >= 31622.78 nM T26500 C2DF8K 57328211 Ki >= 31622.78 nM T26500 C0QDE3 57328212 Ki >= 31622.78 nM T26500 CS25HQ 57328213 Ki >= 31622.78 nM T26500 CR1L2W 57328276 Ki >= 31622.78 nM T26500 CFE9O8 57328277 Ki >= 31622.78 nM T26500 C6Z4IJ 57390145 Ki = 5080 nM T26500 C0P9VG 57390224 Ki = 15848.93 nM T26500 CBD1F0 57390225 Ki = 27542.29 nM T26500 C96MYC 57390262 Ki = 613 nM T26500 C5TC9G 57390263 Ki = 139 nM T26500 C5TG6E 57390264 Ki > 10000 nM T26500 CF86RJ 57390344 Ki > 2000 nM T26500 CE84NL 57391032 Ki = 104 nM T26500 CRS02A 57391033 Ki = 145 nM T26500 CE0I6C 57391034 Ki = 155 nM T26500 CB62SR 57391122 Ki = 20000 nM T26500 C6ZF3E 57391128 Ki > 10000 nM T26500 CPK4B9 57391129 Ki > 205 nM T26500 CY07AU 57391819 Ki = 15 nM T26500 CZ20EU 57391926 Ki = 102 nM T26500 C9B5CM 57391927 Ki = 2670 nM T26500 CBJ6X8 57391928 Ki = 2090 nM T26500 CAL75E 57392460 Ki = 1995.26 nM T26500 CP5O1Y 57392827 Ki = 13 nM T26500 CUJ7C2 57392889 Ki = 34900 nM T26500 C3YV7C 57392890 Ki > 2000 nM T26500 C4O3FM 57393651 Ki = 973 nM T26500 CXV65K 57393730 Ki = 10471.29 nM T26500 CMAB34 57393768 Ki > 10000 nM T26500 C8UA6K 57393769 Ki = 196 nM T26500 CJOX95 57393770 Ki = 443 nM T26500 COCA67 57393771 Ki = 416 nM T26500 CR7E2U 57393772 Ki = 3227 nM T26500 C3V9JZ 57393773 Ki = 33 nM T26500 CU7ZE2 57393774 Ki = 35 nM T26500 CHYX48 57394548 Ki = 21 nM T26500 CB96GL 57394549 Ki = 26 nM T26500 C5AK4C 57394550 Ki = 180 nM T26500 C4OS6L 57394625 Ki = 1600 nM T26500 CZSU79 57394626 Ki = 939 nM T26500 C7GY8V 57394627 Ki = 593 nM T26500 C5CA6U 57394628 Ki = 201 nM T26500 CW7R1K 57394636 Ki = 53 nM T26500 C3G5XA 57394637 Ki > 10000 nM T26500 CUS6C8 57395260 Ki = 649 nM T26500 CAC10J 57395494 Ki = 884 nM T26500 C9SGJ4 57395495 Ki > 10000 nM T26500 CS16IR 57395496 Ki = 272 nM T26500 CG83KQ 57395497 Ki > 10000 nM T26500 CMQ17F 57395498 Ki > 10000 nM T26500 CICN31 57395499 Ki = 885 nM T26500 CF4A6M 57395538 Ki = 53 nM T26500 C5HEN8 57395619 Ki = 212 nM T26500 CI5M2U 57395620 Ki = 502 nM T26500 CY6BP7 57395916 IC50 > 10000 nM T26500 CY07ZQ 57396298 Ki = 21 nM T26500 C9SE1H 57396299 Ki = 156 nM T26500 CKWY43 57396300 Ki = 156 nM T26500 C1U7YK 57396301 Ki = 1 nM T26500 CJ5Q6X 57396382 Ki = 20000 nM T26500 CE3U5Q 57397301 Ki = 6760.83 nM T26500 CY87IN 57397738 Ki > 20000 nM T26500 C69ABZ 57398091 Ki = 7.7 nM T26500 C0IN2H 57398176 Ki = 860 nM T26500 CC9X4Z 57398182 Ki > 10000 nM T26500 C7U8TI 57398183 Ki = 46 nM T26500 C6N4KZ 57398985 Ki = 14125.38 nM T26500 CLE0O5 57399016 Ki = 837 nM T26500 CQ0BO9 57399017 Ki > 10000 nM T26500 CK8VN0 57399018 Ki = 37 nM T26500 CBM57H 57399019 Ki = 376 nM T26500 CDW12V 57399107 Ki = 2110 nM T26500 CR25WT 57399746 Ki = 0.8 nM T26500 CFG2A8 57399747 Ki = 39 nM T26500 CL3G2O 57399827 Ki = 235 nM T26500 CZ12OJ 57399828 Ki = 601 nM T26500 CH90TP 57399829 Ki = 32.4 nM T26500 C0BXZ6 57400473 Ki = 676 nM T26500 C1F8MJ 57400589 Ki = 83 nM T26500 C04XQW 57400700 Ki = 22387.21 nM T26500 CK6TI8 57400735 Ki = 42 nM T26500 CKH87Z 57400736 Ki > 10000 nM T26500 CP14NT 57400737 Ki = 882 nM T26500 CT2C7A 57400738 Ki = 16 nM T26500 CP75KQ 57400777 Ki = 16 nM T26500 C06WSZ 57400778 Ki = 39 nM T26500 COB2Q3 57401167 Ki = 74 nM T26500 C6OL8I 57401517 Ki = 7.7 nM T26500 CV7UN2 57401602 Ki = 930 nM T26500 CQ5XE0 57401609 Ki > 10000 nM T26500 C4RN6L 57402471 Ki = 5888.44 nM T26500 C6PH5T 57402472 Ki = 8912.51 nM T26500 C6T4LQ 57402512 Ki = 250 nM T26500 C8V4ZA 57402513 Ki > 10000 nM T26500 CVK01R 57402514 Ki = 346 nM T26500 C10PXB 57402928 Ki = 3170 nM T26500 C8ZMQ2 57402929 Ki = 129 nM T26500 CQ7O6B 57403269 Ki = 1280 nM T26500 C1JFL4 57403350 Ki = 23.6 nM T26500 CM2UK4 57403351 Ki = 58.9 nM T26500 C4RHF3 57404027 Ki > 10000 nM T26500 CUOV05 57411066 Ki > 10000 nM T26500 C46RXK 58227085 Ki = 45 nM T26500 C3I2AT 58227086 Ki = 5 nM T26500 C5XDA0 58227127 Ki = 63 nM T26500 C8HQ0I 58227143 Ki = 55 nM T26500 C0Y6CW 58227144 Ki = 365 nM T26500 C0Y3MG 58227148 Ki = 0.8 nM T26500 CZI13T 58227157 Ki = 6 nM T26500 C74FMS 58227158 Ki = 10000 nM T26500 C3Y8RI 58227165 EC50 = 112 nM T26500 CZWU37 58227179 Ki = 8 nM T26500 CG92LX 58227200 Ki = 6 nM T26500 C9W8CM 58227207 Ki = 389 nM T26500 C2BPY8 58227216 Ki = 240 nM T26500 CAX85N 58227242 Ki = 824 nM T26500 C7Z9UX 58227252 Ki = 2 nM T26500 C3SN0G 58227255 Ki = 2 nM T26500 CJV95A 58227259 Ki = 8 nM T26500 CJ5R2U 58227260 EC50 = 20 nM T26500 C4D5PZ 58227319 Ki = 134 nM T26500 CNOU75 58227326 Ki = 3 nM T26500 CGI87R 58227337 Ki = 6 nM T26500 CBED65 58227340 Ki = 4 nM T26500 CQX5N4 58227342 Ki = 1 nM T26500 C5S0ZW 58227388 Ki = 69 nM T26500 C0YWT1 58509213 IC50 > 10000 nM T26500 CYKF93 59651916 Ki > 10000 nM T26500 C0JFX7 59777258 Ki = 2.9 nM T26500 CQAR42 59777262 Ki = 36 nM T26500 CZ14TI 59777309 Ki = 159 nM T26500 C9PYK5 59777338 Ki = 0.92 nM T26500 C5KCZ6 59777341 Ki = 2.3 nM T26500 CSNZ26 60150162 Ki = 3235.94 nM T26500 C9YP3F 60150166 Ki = 1202.26 nM T26500 CNG8B4 63868018 Ki = 2664 nM T26500 CN85KQ 63868172 Ki = 812 nM T26500 CPJ2C1 63868328 Ki = 185 nM T26500 C9DKI0 66572102 Ki = 3981.07 nM T26500 C03ZTD 66572103 Ki = 6309.57 nM T26500 C5AWB7 66572104 Ki = 1995.26 nM T26500 CWY2G9 66572105 Ki = 31.62 nM T26500 CD48KZ 66572106 Ki = 31.62 nM T26500 C1I8GV 66572107 Ki = 1000 nM T26500 CD6U3T 66572108 Ki = 158.49 nM T26500 CMQ8U1 66572109 Ki = 794.33 nM T26500 CNE65V 66572110 Ki = 5011.87 nM T26500 C2ZP1D 66572111 Ki = 12589.25 nM T26500 CR67CU 66572112 Ki = 1995.26 nM T26500 CH4DJ5 66572113 Ki = 79.43 nM T26500 CTU65J 66572114 Ki = 19.95 nM T26500 CQ5IJ9 66572115 Ki = 1000 nM T26500 CF6AC8 66572116 Ki = 39.81 nM T26500 C7H2TE 66573456 Ki = 398.11 nM T26500 CNSR56 66573457 Ki = 79.43 nM T26500 C64GCV 66573458 Ki = 6.31 nM T26500 CDT3L8 66573459 Ki = 6.31 nM T26500 C1QD2Z 66573460 Ki = 12.59 nM T26500 CCN86U 66573462 Ki = 199.53 nM T26500 C8E5SI 66573463 Ki = 31.62 nM T26500 CO14JR 66740470 Ki = 56 nM T26500 CKXB42 66740859 Ki = 1.7 nM T26500 CH4T3U 66740898 Ki = 25 nM T26500 CH54BP 66741667 Ki = 520 nM T26500 COZ23Y 67087450 Ki = 55 nM T26500 CF9SX7 68081305 Ki = 20 nM T26500 C0QIS3 68081433 Ki = 39 nM T26500 C9O8ED 70681961 Ki = 39.81 nM T26500 CM75RW 70681962 Ki = 63.1 nM T26500 CU2O5S 70681963 Ki = 15.85 nM T26500 CQ2G7Z 70684084 Ki = 251.19 nM T26500 COG3X0 70684085 Ki = 5011.87 nM T26500 C5U4TO 70686222 Ki = 501.19 nM T26500 CBUR71 70686223 Ki = 398.11 nM T26500 C1AOQ6 70686224 Ki = 251.19 nM T26500 C9W2VZ 70688339 Ki = 63.1 nM T26500 CG9RZ5 70688340 Ki = 79.43 nM T26500 CVH14D 70690367 Ki = 15848.93 nM T26500 C96MXB 70690368 Ki = 1584.89 nM T26500 C58ADF 70690369 Ki = 19.95 nM T26500 C8ZM3L 70692528 Ki = 251.19 nM T26500 CY97BC 70692529 Ki = 10 nM T26500 CIP5Y1 70692530 Ki = 398.11 nM T26500 C6XP2O 70692531 Ki = 39.81 nM T26500 CURD51 70694582 Ki = 398.11 nM T26500 C07TMA 70696620 Ki = 5.012 nM T26500 C5YZ2J 70696621 Ki = 39.81 nM T26500 C78KCG 70696622 Ki = 31.62 nM T26500 CBM4O2 70696623 Ki = 100 nM T26500 CE6YD5 71450707 Ki > 10000 nM T26500 C4X9KY 71454294 Ki > 10000 nM T26500 CA65OQ 71454295 Ki > 10000 nM T26500 CD4HQ6 71456045 Ki > 10000 nM T26500 CD78KL 71456046 Ki > 10000 nM T26500 CSX5J0 71457844 Ki > 10000 nM T26500 CD10CQ 71459761 Ki > 1000 nM T26500 CE9H8S 71461658 Ki = 244 nM T26500 C2AI5H 71518535 Ki = 10450 nM T26500 CL5SI6 71518536 Ki = 2670 nM T26500 CJ4EX3 71518698 Ki = 45920 nM T26500 C7NG1P 71518859 Ki = 1410 nM T26500 C1S9GF 71518860 Ki = 5400 nM T26500 CR91GC 71518861 Ki = 2640 nM T26500 CVET73 71518862 Ki = 3280 nM T26500 C2C0SN 71518863 Ki = 3320 nM T26500 CB2F9O 71518864 Ki = 3730 nM T26500 C0UP8F 71518865 Ki = 7320 nM T26500 CYS80T 71519010 Ki = 8990 nM T26500 CZV9W5 71519011 Ki = 36120 nM T26500 CM7VD9 71519012 Ki = 390 nM T26500 C92MOP 71519013 Ki = 4070 nM T26500 CB3FY1 71519014 Ki = 48010 nM T26500 CM8LD0 71519015 Ki = 8720 nM T26500 CRA8K3 71519016 Ki = 1410 nM T26500 C12ITS 71519176 Ki = 2930 nM T26500 CC8A1M 71519177 Ki = 1710 nM T26500 CIZ5O9 71519178 Ki = 980 nM T26500 CDLO59 71519179 Ki = 5950 nM T26500 CB2GV4 71519346 Ki = 36350 nM T26500 CVE2T8 71519347 Ki = 8130 nM T26500 C9HR2Y 71519348 Ki = 25220 nM T26500 CBF5Y8 71519349 Ki = 44150 nM T26500 C4JX6C 71519499 Ki = 67870 nM T26500 C7E6CY 71519500 Ki > 100000 nM T26500 CLQ31I 71519674 Ki = 5.248 nM T26500 C8JC6A 71525586 Ki = 9.333 nM T26500 CR9ZE5 71525587 Ki = 53.7 nM T26500 CRL42M 71525588 Ki = 25.12 nM T26500 CZ0FT2 71525589 Ki = 12.3 nM T26500 CRM9Q1 71525678 Ki = 10.72 nM T26500 C2GK7O 71525679 Ki = 9.12 nM T26500 C7HR1A 71525680 Ki = 10.23 nM T26500 C8A0NC 71525681 Ki = 6.457 nM T26500 CE92DF 71528209 Ki = 7476 nM T26500 C5RK1W 71551636 Ki = 3.162 nM T26500 C3XKL2 71603135 Ki = 12.3 nM T26500 CQ3Y9W 71603136 Ki = 3.388 nM T26500 CT8WF0 71603137 Ki = 35.48 nM T26500 CDW08C 71603138 Ki = 15.14 nM T26500 CA4GQ7 71603139 Ki = 11.48 nM T26500 CK4T5Q 71603140 Ki = 7.079 nM T26500 C70OBY 71603141 Ki = 14.79 nM T26500 C1HEY4 71603142 Ki = 11.22 nM T26500 CUW27Q 71603194 Ki = 16.98 nM T26500 CO2P7E 71603195 Ki = 21.88 nM T26500 CX3JY7 71681474 Ki = 794.33 nM T26500 CW7GI6 71681475 Ki = 79.43 nM T26500 CCR0K8 71681476 Ki = 25.12 nM T26500 COA15E 71681477 Ki = 1000 nM T26500 CH1QS5 71681478 Ki = 398.11 nM T26500 C9WR5O 71681479 Ki = 3162.28 nM T26500 C9QG3Z 71681480 Ki = 1995.26 nM T26500 C59VTX 71681639 Ki = 39.81 nM T26500 C74NFK 71681640 Ki = 2511.89 nM T26500 CI0YL4 71681641 Ki = 630.96 nM T26500 CZ2W4R 71681642 Ki = 1258.93 nM T26500 CRQ48M 71681643 Ki = 79.43 nM T26500 CWFV56 71681644 Ki = 50.12 nM T26500 CA53YR 71681645 Ki = 79.43 nM T26500 C8UW7T 71681802 Ki = 1000 nM T26500 C6NZV9 71681803 Ki = 501.19 nM T26500 CI6YF8 71681804 Ki = 10 nM T26500 CJU7R2 71681805 Ki = 50.12 nM T26500 CSN26Z 71681806 Ki = 39.81 nM T26500 C5SV0C 71681807 Ki = 10 nM T26500 C5TUB8 71681808 Ki = 31.62 nM T26500 C84RTX 71681974 Ki = 79.43 nM T26500 CPM9J0 71681975 Ki = 1258.93 nM T26500 CIFN53 71681976 Ki = 316.23 nM T26500 CC5B3R 71681977 Ki = 3162.28 nM T26500 CB1A5V 71681978 Ki = 10000 nM T26500 C93WIJ 71712245 Ki = 1412537.54 nM T26500 CW5MC4 71717291 Ki = 316.23 nM T26500 CC6Q5R 72771081 Ki < 100 nM T26500 CG4V9Q 73346048 Ki = 6760.83 nM T26500 CMJ6R2 73347579 Ki > 100000 nM T26500 C7E1KJ 73347580 Ki > 100000 nM T26500 CY60RD 73347826 Ki > 10000 nM T26500 C9MW8L 73353369 Ki = 30.9 nM T26500 CH2BZ4 73355143 Ki = 16218.1 nM T26500 C4S7TA 76311195 Ki = 5.012 nM T26500 C8CE2R 76313483 Ki > 1000 nM T26500 CU8CX7 76314798 Ki = 7.943 nM T26500 C98BJM 90643887 IC50 > 10000 nM T26500 CP68KJ 90645145 Ki = 520 nM T26500 C8R2BY 90645146 Ki = 378 nM T26500 C3U1IQ 90645147 Ki = 203 nM T26500 C6GP1L 90645148 Ki = 5161 nM T26500 CR4S1U 90645149 Ki = 1747 nM T26500 CB8FN4 90645150 Ki = 408 nM T26500 C6W4BT 90645151 Ki = 1261 nM T26500 CJ79LD 90645152 Ki = 2391 nM T26500 C1ETP7 90645153 Ki = 431 nM T26500 CG47OW 90645154 Ki = 4239 nM T26500 C6UO1G 90645155 Ki = 2358 nM T26500 CML3K8 90645156 Ki = 64490 nM T26500 CSY2C4 90645157 Ki = 1472 nM T26500 C8F4SL 90645158 Ki = 6007 nM T26500 CJR5A7 90645159 Ki = 790 nM T26500 CCWN73 90645160 Ki = 5077 nM T26500 C95FIW 90645161 Ki = 1191 nM T26500 C9SL1H 90645162 Ki = 1787 nM T26500 C3AK8Z 90645163 Ki = 10567 nM T26500 CES65T 90645164 Ki = 834 nM T26500 CF05GE 90654501 Ki = 20417.38 nM T26500 C1BJC6 90654502 Ki = 331131.12 nM T26500 CPY4X2 90654503 Ki = 9332.54 nM T26500 C1TSD9 90655027 Ki = 25 nM T26500 CE93KU 90655028 Ki = 36 nM T26500 CUL3A8 90655029 Ki = 328 nM T26500 C7N5QF 90655030 Ki > 10000 nM T26500 CV41DQ 90655031 Ki > 10000 nM T26500 CZ4Y3V 90667228 EC50 = 2884.03 nM T26500 CGWN45 90667229 EC50 = 776.25 nM T26500 CT4WV7 90667238 EC50 = 549.54 nM T26500 C96AHZ 90667239 EC50 = 467.74 nM T26500 CMUX10 90667240 EC50 = 245.47 nM T26500 C8FXR0 90667434 EC50 = 1000 nM T26500 CFA3D4 112936251 EC50 = 912.01 nM T26500 C85IFK 112936262 Ki = 1737.8 nM T26500 CLQ10U 112936267 Ki = 9772.37 nM T26500 C5DU3L 112936341 Ki = 31622.78 nM T26500 C1LO3K 112936352 Ki = 72443.6 nM T26500 CI0DB6 112936357 Ki = 36307.81 nM T26500 CBT56P 117724523 Ki = 7 nM T26500 C7Y5AL 118720433 Ki = 456 nM T26500 CD5TF8 118720434 Ki = 92 nM T26500 C5YUK9 118720435 Ki = 126 nM T26500 CW5KE8 118720436 Ki > 10000 nM T26500 CT7C3H 118720437 Ki = 11 nM T26500 CN91FO 118720438 Ki = 460 nM T26500 CQO1Y5 118720439 Ki = 1547 nM T26500 CQ4GW1 118720440 Ki > 1000 nM T26500 CZ03GM 118720441 Ki = 50 nM T26500 C3J6YN 118720442 Ki = 2 nM T26500 CZ7Y0I 118720443 Ki > 10000 nM T26500 CE74UX 118725538 Ki = 216 nM T26500 C0T5KZ 118725539 Ki = 142 nM T26500 C0H7UQ 118725540 Ki = 97 nM T26500 C4IM3V 118725541 Ki = 176 nM T26500 CW13SQ 118725542 Ki = 118 nM T26500 C4G3YC 118734875 Ki > 10000 nM T26500 C9AIE1 118734876 Ki > 10000 nM T26500 CNF47H 121238066 Ki = 14610 nM T26500 CQ26TZ 121238067 Ki = 529 nM T26500 CWU1A0 121238068 Ki = 5600 nM T26500 C8I7TE 121238069 Ki = 7499 nM T26500 C6KO5C 121238070 Ki = 10610 nM T26500 C0KO2A 121238071 Ki = 3190 nM T26500 CPVZ72 122193094 Ki = 4860 nM T26500 C9D6BC 122193095 Ki = 253 nM T26500 CPYT06 122193096 Ki = 4210 nM T26500 C95SBK 122193097 Ki = 9040 nM T26500 CO2B6D 122193098 Ki = 1780 nM T26500 C1QMG9 122193099 Ki = 1140 nM T26500 CB39GI 122193100 Ki = 3520 nM T26500 C64DPA 122193101 Ki = 2450 nM T26500 C7SR4T 122193102 Ki = 2640 nM T26500 CP5N0J 122193103 Ki = 2570 nM T26500 CD7J9K 122193104 Ki = 29985 nM T26500 CN1LS6 122193105 Ki = 3794 nM T26500 CQG95C 122193106 Ki = 2525 nM T26500 CB7S4V 122194623 Ki = 5210 nM T26500 CVI17K 122194624 Ki = 2230 nM T26500 C45OUD 122194625 IC50 = 606 nM T26500 CI84EH 122194626 Ki = 37400 nM T26500 CK61AT 127026016 Ki = 26302.68 nM T26500 C9LJH1 127026017 Ki = 13803.84 nM T26500 C3QBS9 127026018 Ki = 6760.83 nM T26500 CDF56P 127026019 Ki = 7762.47 nM T26500 C0Z9RT 127035835 EC50 = 933.25 nM T26500 C20IYZ 127035836 Ki = 19952.62 nM T26500 CL9PN3 127035837 Ki = 10964.78 nM T26500 CST95G 127036978 Ki = 4265.8 nM T26500 CIK1S7 127036979 Ki = 9120.11 nM T26500 C1ICF6 127036980 Ki = 14454.4 nM T26500 CP6IZ7 127036981 Ki = 15135.61 nM T26500 CY6T9R 127036982 Ki = 19498.45 nM T26500 C4KO0Z 127048828 EC50 = 15 nM T26500 C2XT3K 127048890 EC50 = 150 nM T26500 CY38PR 127049156 EC50 = 230 nM T26500 CG35RK 127049855 EC50 = 500 nM T26500 C5BZ6T 127049856 Ki = 290 nM T26500 CT9SP3 127050018 Ki = 354.81 nM T26500 CVEK19 127050019 Ki = 158.49 nM T26500 CZMO27 127050309 Ki = 3.388 nM T26500 CRUY19 127050310 Ki = 1 nM T26500 CF0Y6S 127050431 EC50 = 111 nM T26500 C6F2RA 127050434 EC50 = 44 nM T26500 C5P1EB 127050776 Ki = 870 nM T26500 CH8G4Z 127051047 EC50 = 2675 nM T26500 CH8Y7R 127051301 EC50 = 63 nM T26500 CB25IM 127051958 EC50 = 1710 nM T26500 CNR4Q9 127051986 EC50 = 125 nM T26500 C3YSF2 127052292 EC50 = 372 nM T26500 C9OSN3 127052293 EC50 = 11 nM T26500 C3WA2L 127052294 EC50 = 129 nM T26500 CYWZ45 127052295 EC50 = 524 nM T26500 C98YAI 127052634 EC50 = 245 nM T26500 C7T4VH 127052635 EC50 = 202 nM T26500 CAVB41 132584404 Ki > 10000 nM T26500 CBU81N 134149168 Ki > 10000 nM T26500 C01XKD 135421235 Ki < 10000 nM T26500 CZT84E 135502653 Ki < 10000 nM T26500 CHSN19 135525668 Ki = 9.5 nM T26500 CJW1V9 135570464 Ki = 15135.61 nM T26500 C7U6ET 135589846 Ki = 4677.35 nM T26500 CL83IO 136016345 Ki = 219 nM T26500 CBS93O 136030655 Ki = 31.62 nM T26500 CZJ9I1 136042265 Ki = 26 nM T26500 C3U6CW 136042266 Ki = 4.6 nM T26500 C8KW7F 136042267 Ki = 24 nM T26500 CFC17Q 136042268 Ki = 4.6 nM T26500 CN5B6D 136042269 Ki = 20 nM T26500 CH9J5X 136042270 Ki = 6.5 nM T26500 C8I7CO 136141537 Ki = 50.12 nM T26500 CRH19Y 136192874 Ki = 15.85 nM T26500 C56FVS 136192886 Ki = 50.12 nM T26500 CH85GS 136773074 Ki = 6750 nM T26500 CI8NR9 137632569 Ki = 3 nM T26500 C4XEF0 137634349 Ki = 16400 nM T26500 CX35KM 137634777 Ki = 3018 nM T26500 C6UVO3 137640214 Ki = 400 nM T26500 C2HMK4 137646103 Ki = 62 nM T26500 C9M8JR 137646744 Ki = 174 nM T26500 CPG0V2 137646939 Ki = 19 nM T26500 COGK52 137647794 Ki = 4200 nM T26500 C7BOY5 137650793 Ki = 3100 nM T26500 C7CM5W 137655927 Ki = 14.5 nM T26500 CWO0B6 137657169 Ki = 2.7 nM T26500 C5F8AB 137658819 Ki = 3800 nM T26500 C8M2UW 137659490 Ki = 4 nM T26500 C6P3SR 153287553 Ki > 10000 nM T26500 CV9G7Z 153287572 Ki > 10000 nM T26500 CO85KL 153287574 Ki > 10000 nM T26500 CLC7N6 155511939 Ki > 10000 nM T26500 CR8M5G 155512115 Ki > 1000 nM T26500 CGAP59 155512724 EC50 = 29.51 nM T26500 C20UBG 155513611 EC50 = 1.905 nM T26500 CN5VE4 155513723 Ki > 10000 nM T26500 CMZ4Q7 155515478 EC50 = 3.162 nM T26500 CTZL14 155516421 EC50 = 0.6026 nM T26500 CGO36Z 155517879 EC50 = 35.48 nM T26500 CVQS21 155518359 Ki > 10000 nM T26500 CUSA24 155519891 Ki > 10000 nM T26500 CM4TF8 155522043 Ki > 10000 nM T26500 CI2Z8F 155524114 EC50 = 0.123 nM T26500 CQS1N5 155525278 EC50 = 3.548 nM T26500 CR52CO 155530956 Ki > 1000 nM T26500 CD4F1G 155531771 Ki > 10000 nM T26500 CR70SX 155533943 Ki > 1000 nM T26500 C8XG9P 155534518 Ki = 446.68 nM T26500 CNK51Q 155535097 Ki = 2691.53 nM T26500 CC9J6W 155535840 Ki > 1000 nM T26500 CB79ZW 155536080 Ki > 10000 nM T26500 CRI5F4 155536508 Ki = 204.17 nM T26500 CCB1A2 155537946 Ki > 1000 nM T26500 CQ02MZ 155538072 Ki > 1000 nM T26500 CM9VU3 155538173 Ki > 10000 nM T26500 CYA2O8 155538400 Ki > 10000 nM T26500 C6QN1S 155538988 Ki = 1905.46 nM T26500 CI37OT 155539096 Ki = 186.21 nM T26500 C3YW8J 155539458 Ki = 354.81 nM T26500 C5E6AH 155539562 Ki = 2847 nM T26500 COF72J 155540201 Ki = 1071.52 nM T26500 CQL0O8 155540438 IC50 = 32 nM T26500 CHQ7A8 155541279 Ki = 13.18 nM T26500 C4OAN9 155543351 Ki > 10000 nM T26500 CZT91D 155543973 Ki > 10000 nM T26500 C1OG6N 155544052 Ki > 10000 nM T26500 C6IO5C 155545099 Ki > 10000 nM T26500 CAY2P0 155545717 Ki = 295 nM T26500 CBQ9C6 155546701 Ki = 247 nM T26500 CO2J0Z 155546798 Ki = 114.82 nM T26500 C1T0BF 155549318 Ki = 2630.27 nM T26500 C29BAV 155550731 Ki = 19900 nM T26500 C7WO9P 155552060 EC50 = 19.5 nM T26500 CZQW48 155552101 Ki = 616.6 nM T26500 CLK7U1 155552340 Ki = 309.03 nM T26500 C7DM5X 155552772 Ki > 1000 nM T26500 C8BVH4 155553066 Ki > 10000 nM T26500 C1RLI0 155553370 Ki > 100000 nM T26500 CF7K5M 155556721 Ki = 470 nM T26500 C6Q2YJ 155558288 Ki > 10000 nM T26500 CJT90H 155558487 Ki > 10000 nM T26500 C5BAG2 155559502 Ki > 10000 nM T26500 C57DRK 155560636 Ki > 10000 nM T26500 CJ2S0E 155563066 Ki > 10000 nM T26500 CJQ59S 155563181 IC50 = 1400 nM T26500 CLC7W8 155563295 Ki > 10000 nM T26500 CR91TB 155563489 Ki = 725 nM T26500 C8HR4Q 155567029 Ki = 21800 nM T26500 C8KY4O 155567055 Ki > 1000 nM T26500 CHD6C8 155567107 Ki = 204.17 nM T26500 C3Q9EC 155568016 Ki = 1331 nM T26500 C5G3FT 155568977 Ki = 166 nM T26500 CP9TR0 10324985 Ki > 10000 nM T26500 D00HWF 6421522 Ki = 50.12 nM T26500 D00XJR 10446295 Ki = 20 nM T26500 D01CJZ 10330240 EC50 < 10000 nM T26500 D01JXM 46222048 Ki = 1.1 nM T26500 D02RAN 3692 Ki = 1.6 nM T26500 D02SQF 37463 EC50 = 31.62 nM T26500 D03SAM 156615 Ki = 146 nM T26500 D03SNI 24759623 Ki = 39.81 nM T26500 D05RGW 11313837 Ki = 1995.26 nM T26500 D06RNM 3032915 EC50 = 19.95 nM T26500 D08BLM 46228160 Ki = 14300 nM T26500 D08BSG 132937 Ki = 12.59 nM T26500 D08DOG 25130235 Ki = 34.67 nM T26500 D08ECP 912 Ki = 316.23 nM T26500 D09ROG 2994072 Ki > 10000 nM T26500 D09RPR 16737207 Ki > 10000 nM T26500 D09WQL 9989505 Ki = 245.47 nM T26500 D0A4XL 3614 Ki = 11000 nM T26500 D0B4SF 41376 Ki = 12.3 nM T26500 D0C8IB 10680721 Ki = 290 nM T26500 D0E5EB 9793868 Ki = 251.19 nM T26500 D0E5XM 13499360 Ki = 10 nM T26500 D0E9SR 4908365 Ki = 3.311 nM T26500 D0F9QT 44538833 Ki = 6 nM T26500 D0G2BS 5013 Ki = 6918.31 nM T26500 D0G3RN 11301441 Ki = 5.623 nM T26500 D0G3RZ 46228161 Ki = 15600 nM T26500 D0G6AQ 23786499 Ki = 1584.89 nM T26500 D0H2KD 921599 Ki = 38 nM T26500 D0H3DY 10374457 EC50 > 0.0001 nM T26500 D0H4TP 9798547 Ki > 3162.28 nM T26500 D0I3XA 6422124 Ki = 612 nM T26500 D0I5CT 126688 Ki = 5011.87 nM T26500 D0K8DZ 11672774 Ki = 501.19 nM T26500 D0KK4C 10154137 EC50 > 0.0001 nM T26500 D0L5MW 181743 Ki > 10000 nM T26500 D0M9IC 441082 Ki > 10000 nM T26500 D0MP8E 3063228 Ki = 25.12 nM T26500 D0O3NG 3077 Ki = 90 nM T26500 D0OM9G 3035842 EC50 = 15.85 nM T26500 D0P8DW 25068753 Ki = 4.677 nM T26500 D0Q2GP 10381810 EC50 = 28.18 nM T26500 D0Q8BS 6603865 Ki = 3981.07 nM T26500 D0Q8NO 10176414 Ki = 10 nM T26500 D0QT2F 756701 Ki = 18400 nM T26500 D0S0HT 9812843 Ki = 100 nM T26500 D0SQ0T 10942498 EC50 > 0.0001 nM T26500 D0T8OD 2790 Ki = 1 nM T26500 D0TC5E 91613 Ki = 794.33 nM T26500 D0U1DR 11492393 Ki = 39.81 nM T26500 D0UK0F 753256 Ki = 290 nM T26500 D0W7OR 9877454 Ki = 4570.88 nM T26851 CM86EA 25082538 IC50 = 12000 nM T26851 C3G6XR 44388600 IC50 = 53600 nM T26851 CV9RB8 44388652 IC50 = 47800 nM T26851 C3P0EW 44388714 IC50 > 1000000 nM T26851 CP83MA 44388727 IC50 > 1000000 nM T26851 CY9W1M 44445329 IC50 = 1200 nM T26851 CN8LQ4 73348620 IC50 = 1500 nM T26851 C07ZGV 73350198 IC50 = 1100 nM T26851 C7E3VK 118730530 IC50 = 4000 nM T26851 C7LT9V 145985080 IC50 = 62 nM T26851 D03SHO 44388602 IC50 = 13000 nM T34064 D00PEH 135449332 Ki = 8480 nM T34064 D02RQU 54687 Ki = 180000 nM T34064 D02ZTJ 5339 Ki = 3000 nM T34064 D07IQS 148192 Ki = 5100 nM T34064 D07POC 176870 Ki = 530 nM T34064 D07VLY 31703 Ki = 230000 nM T34064 D0AZ8C 5213 IC50 = 4500 nM T34064 D0G3DL 135398735 Ki = 63000 nM T34064 D0R1RS 3715 Ki = 130000 nM T34064 D0ZU9R 392622 Ki = 5900 nM T34064 D0C5VQ 1548994 IC50 = 800 nM T34064 D0G7UX 5284373 Ki = 36000 nM T34064 C4J5ZF 185617 Ki = 25900 nM T34064 CNI9X4 5281888 Ki = 2800 nM T34064 CM47KI 5351344 IC50 = 12270 nM T34064 CI28JY 10457775 IC50 > 200000 nM T34064 C47ZJY 11996857 Ki = 25900 nM T34064 D0G2JZ 1464 Ki = 20000 nM T79031 D07EXH 359 IC50 = 36470 nM T79031 D08SKH 4114 IC50 > 500000 nM T79031 D09EGZ 2719 IC50 = 7000 nM T79031 D09XZB 123631 IC50 = 20000 nM T79031 D0K8KX 5280343 IC50 = 5400 nM T79031 D0NS6H 3152 IC50 = 240 nM T79031 D00VUI 6199 IC50 > 500000 nM T79031 D00XKB 57406537 IC50 = 0.2 nM T79031 D01AYX 57404290 IC50 = 0.28 nM T79031 D04OSA 46202416 IC50 = 0.6 nM T79031 D07SDQ 969516 IC50 = 343000 nM T79031 D08MHD 57827330 IC50 = 7 nM T79031 D0CG8S 71305058 IC50 = 2 nM T79031 D0F8GK 49837968 IC50 = 12 nM T79031 D0H6AG 51003469 IC50 = 4 nM T79031 D0N1BF 44251605 IC50 = 240 nM T79031 D0O8UB 53241828 IC50 = 21 nM T79031 D0QR5G 2355 IC50 > 500000 nM T79031 D0R4KK 51352361 IC50 = 0.4 nM T79031 D0T7BV 60202321 IC50 = 5.5 nM T79031 D0U2BH 65064 IC50 = 757 nM T79031 D0Y0EP 67979346 IC50 = 0.2 nM T79031 D0Y5NA 118435360 IC50 = 5 nM T79031 D0E3SX 23627211 Ki = 7.8 nM T79031 D03OLC 11359820 Ki = 530 nM T79031 D0H4IY 59262421 Ki = 99 nM T79031 D0QX1S 11581511 Ki = 190 nM T79031 D0RN2X 442126 IC50 > 500000 nM T79031 C5ECM1 3651 IC50 > 100000 nM T79031 C2ESO4 8417 IC50 > 500000 nM T79031 CU7FA5 10211 Ki = 6200 nM T79031 CV24FH 10228 IC50 > 500000 nM T79031 C8IWZ0 10236 IC50 = 776000 nM T79031 C5SRE2 10658 IC50 > 500000 nM T79031 C3W0JR 11379 IC50 = 2000000 nM T79031 CBI9W2 17536 IC50 > 500000 nM T79031 C9ZO6A 21527 IC50 = 731000 nM T79031 CPV3D9 33306 IC50 = 359200 nM T79031 CBP71W 65056 IC50 = 4500 nM T79031 CX4FN2 65084 IC50 = 2500 nM T79031 C1FD4A 65090 IC50 > 500000 nM T79031 C1NQ8E 65188 IC50 > 500000 nM T79031 C0CIP2 65714 IC50 = 6600 nM T79031 CMLI08 68079 IC50 > 500000 nM T79031 C09AHX 68081 IC50 = 244200 nM T79031 C7LF0S 68229 IC50 > 500000 nM T79031 CA0OI5 68486 IC50 > 500000 nM T79031 C09VGT 72859 IC50 = 15960 nM T79031 C2XSU3 73253 IC50 > 500000 nM T79031 C8CQW2 73742 IC50 = 2000000 nM T79031 C2I7WP 74721 IC50 = 2900 nM T79031 C8RYL4 92201 IC50 > 500000 nM T79031 CU7IR2 94727 IC50 = 23260 nM T79031 CZB67X 98608 IC50 = 1432000 nM T79031 CEXR79 160776 IC50 = 5100 nM T79031 C9N0JQ 179897 IC50 > 200000 nM T79031 C5Q1JX 182232 IC50 = 23000 nM T79031 CFZ9X6 206031 Ki = 1.6 nM T79031 CXU5P7 213731 EC50 = 23500 nM T79031 C5JGS7 284056 IC50 = 790000 nM T79031 C5HCA0 296675 IC50 = 9330 nM T79031 CY8NS0 320362 IC50 > 500000 nM T79031 CNP1J9 334704 IC50 > 500000 nM T79031 C4J8FX 340211 IC50 = 180000 nM T79031 C15BDG 341044 IC50 = 1800 nM T79031 CYI84X 442127 IC50 > 500000 nM T79031 C6VC4K 445649 Ki = 1.2 nM T79031 C8NGY9 448772 IC50 = 1400 nM T79031 CY3N2J 449107 IC50 = 500 nM T79031 CJG04U 458010 IC50 = 443600 nM T79031 C5UM8B 513197 IC50 = 27700 nM T79031 C4VI9P 600670 IC50 > 500000 nM T79031 CZ0AH3 638278 IC50 = 51500 nM T79031 C1AH9F 776121 IC50 > 500000 nM T79031 C50NVY 784043 IC50 = 550 nM T79031 C4TAX6 784405 IC50 = 660 nM T79031 C1JUV7 789289 IC50 = 217000 nM T79031 CSO83T 821449 IC50 = 3442000 nM T79031 CIH45J 1018255 IC50 = 1770 nM T79031 CF53LI 1047096 IC50 = 100000 nM T79031 CQ6U2H 1483116 IC50 = 928000 nM T79031 C72CAB 1550607 IC50 = 345100 nM T79031 C4YUX5 1594254 IC50 = 100000 nM T79031 CYV73P 1609819 IC50 = 200000 nM T79031 C96YXL 1717763 IC50 = 50000 nM T79031 CPI20R 1733213 IC50 = 20000 nM T79031 CLW0X5 1796032 IC50 = 500000 nM T79031 CC6L1N 1798772 IC50 = 100000 nM T79031 CKU54M 1826494 IC50 = 100000 nM T79031 C20JZF 1898613 IC50 = 710 nM T79031 CBEC45 2742082 IC50 = 6300 nM T79031 CFY06R 2824823 Ki = 210 nM T79031 CKDJ07 2836198 IC50 = 2990 nM T79031 CY7GM6 2870407 IC50 = 100000 nM T79031 C1VTI0 2908418 IC50 = 3000 nM T79031 CO2K0X 2908827 IC50 = 7100 nM T79031 CI5SD6 2950966 IC50 = 770000 nM T79031 CU17KZ 3055167 IC50 = 104900 nM T79031 C4MZA5 3083726 IC50 > 500000 nM T79031 CC4XV1 3108347 IC50 = 100000 nM T79031 CWSQ93 3122846 IC50 = 2700 nM T79031 CU0QA7 3122847 IC50 = 2600 nM T79031 C7VD2H 3126028 IC50 = 253000 nM T79031 C4ZHE7 3129559 IC50 = 3900 nM T79031 C58NLF 3131985 IC50 = 50000 nM T79031 C5VAE3 3143447 IC50 = 500000 nM T79031 CD3A4I 3285031 IC50 = 2830 nM T79031 C7CKT1 3470183 IC50 = 100000 nM T79031 CSD6V2 3575784 IC50 = 14700 nM T79031 CE3T5B 3718101 IC50 = 100000 nM T79031 C2NJU7 3750579 IC50 = 500000 nM T79031 CX0L8S 3774706 IC50 = 500000 nM T79031 CQ0N9X 3845940 IC50 = 690 nM T79031 CH90DJ 3921980 IC50 = 34500 nM T79031 CT3ZS5 3945434 IC50 = 18000 nM T79031 CCT47S 3948694 IC50 = 97 nM T79031 CN9YC8 3959062 IC50 = 100000 nM T79031 CGO3F0 4014588 IC50 = 1700 nM T79031 CW9US5 4039803 IC50 = 120 nM T79031 CFS84D 4068751 IC50 = 100000 nM T79031 CRE3N6 4088061 IC50 = 100000 nM T79031 CFDC46 4112670 IC50 = 100000 nM T79031 C5U1DO 4131129 IC50 = 100000 nM T79031 C3PY1K 4140894 IC50 = 100000 nM T79031 CBY6K8 4243074 IC50 = 57.8 nM T79031 CR1LX3 4250961 IC50 = 100000 nM T79031 CQV8G3 4253932 IC50 = 10200 nM T79031 C1J3PH 4310580 IC50 = 1000000 nM T79031 CYZ90B 4334360 IC50 = 20000 nM T79031 CL67TU 4338097 IC50 > 50000 nM T79031 CJF16S 4373382 IC50 = 21000 nM T79031 CP4KY6 4415300 IC50 = 90000 nM T79031 CZ47XO 4531891 IC50 = 50000 nM T79031 CLO3Y6 4538151 IC50 = 118000 nM T79031 C9G7KI 4557993 IC50 = 2800 nM T79031 CF2MI7 4561275 IC50 = 2400 nM T79031 CA80KR 4565067 IC50 = 500000 nM T79031 C2CP7Q 4573536 IC50 = 12200 nM T79031 C9EY0N 4599004 IC50 = 100000 nM T79031 CW13EA 4652689 IC50 = 100000 nM T79031 CQ2WS3 4655667 IC50 > 50000 nM T79031 CM90QO 4670102 IC50 = 100000 nM T79031 CAOH69 4789430 IC50 = 9900 nM T79031 CK9AT5 4792504 IC50 = 2000 nM T79031 CDV3O6 4846969 IC50 = 220 nM T79031 C61WHN 4986873 IC50 = 3000 nM T79031 C39YUK 5031416 IC50 = 100000 nM T79031 CWSL73 5040262 Ki = 9400 nM T79031 C2DQT9 5126848 IC50 = 20000 nM T79031 CEH24M 5135855 IC50 = 100000 nM T79031 CLQ2Z6 5162066 IC50 = 100000 nM T79031 C80FTS 5181282 IC50 > 100000 nM T79031 CJ76HG 5214207 IC50 = 2900 nM T79031 C3ZJ8U 5281609 IC50 > 10000 nM T79031 C0D3PO 5281671 IC50 = 59400 nM T79031 CGSC72 5287532 IC50 = 10 nM T79031 COB0W2 5316525 IC50 = 412900 nM T79031 CCWD20 5317564 IC50 = 20400 nM T79031 CPRI38 5320318 IC50 > 500000 nM T79031 C5K0BY 5324473 IC50 = 2540 nM T79031 CZU79V 5327063 IC50 = 98 nM T79031 CQG46M 5376215 IC50 > 500000 nM T79031 COR29P 5469423 IC50 > 5000 nM T79031 CUL7A5 5471349 Ki = 700 nM T79031 CH6DT9 5481958 Ki = 2200 nM T79031 CC6IV0 5481968 IC50 = 135900 nM T79031 CH8AJ6 5481969 IC50 = 101200 nM T79031 CWS5X0 5481970 IC50 = 60600 nM T79031 CMOI48 5481973 IC50 = 146100 nM T79031 C81PIJ 5494406 IC50 = 39 nM T79031 CDG23K 5494410 IC50 = 10 nM T79031 C0KSG2 5494423 Ki = 26 nM T79031 CB05MJ 6405777 IC50 = 100000 nM T79031 C2NVI7 6411782 IC50 = 100000 nM T79031 C0KGW4 6440422 IC50 = 9900 nM T79031 C4GNO1 6442182 IC50 = 11100 nM T79031 CHF7I1 6451462 IC50 = 11430 nM T79031 CRS54N 6540293 Ki = 0.3 nM T79031 C8U5HO 6616205 IC50 = 100000 nM T79031 CC2VX3 6616618 IC50 = 50000 nM T79031 CLT30N 6619193 IC50 = 100000 nM T79031 C6EFT0 6712920 IC50 > 5000 nM T79031 CCJ09A 6918517 Ki = 9.6 nM T79031 COV2Q0 6918701 IC50 = 120 nM T79031 COV50T 6918716 IC50 = 30 nM T79031 C26JWC 6918718 IC50 = 413 nM T79031 C3A6MT 6918719 IC50 = 86 nM T79031 CL3M4K 6918720 IC50 = 91 nM T79031 CGMH34 6918729 IC50 = 45 nM T79031 C4I3CE 6918730 IC50 = 35 nM T79031 CZ2BY9 6918739 IC50 = 16 nM T79031 CD85OL 6918740 IC50 = 4.7 nM T79031 CLK6P7 6918784 IC50 = 8.2 nM T79031 CCO9N0 6918785 IC50 = 3.9 nM T79031 C8P5EL 6918820 Ki = 14 nM T79031 C3OD0J 6918853 IC50 < 10 nM T79031 CR59LJ 9547928 IC50 = 156 nM T79031 CPCN93 9547929 IC50 = 190 nM T79031 C6BPW3 9802458 Ki = 4000 nM T79031 CP9QX2 9808761 IC50 = 130 nM T79031 CA87TI 9809811 IC50 = 50 nM T79031 C08HQG 9832080 IC50 = 281 nM T79031 C4CVL1 9868950 IC50 = 350 nM T79031 CLD37S 9875397 IC50 = 60 nM T79031 CRI0T1 9916309 IC50 = 20 nM T79031 CT1Y4A 9917907 IC50 = 2 nM T79031 CLF04H 9938431 IC50 = 12 nM T79031 CW67YS 9939419 IC50 = 3 nM T79031 CYLG46 9959612 IC50 = 7500 nM T79031 C2P3DU 9983140 IC50 = 180 nM T79031 CIBZ30 9984485 IC50 = 2090 nM T79031 C93KNF 9986236 IC50 = 290 nM T79031 CHG57R 9986500 IC50 = 310 nM T79031 CJ9WA5 10005029 IC50 = 810 nM T79031 C17HZK 10005121 IC50 = 61 nM T79031 C8XV3Y 10008157 IC50 = 40 nM T79031 CJ8B0Q 10028131 IC50 = 127 nM T79031 C5QUJ1 10043694 IC50 > 500000 nM T79031 CEQP27 10049905 IC50 = 46 nM T79031 CN2J9E 10054920 IC50 = 10 nM T79031 CY9SK0 10073810 IC50 = 2450 nM T79031 CEFK38 10077756 IC50 = 190 nM T79031 CAKR94 10077830 IC50 = 11 nM T79031 CJ4TR1 10078059 IC50 = 3 nM T79031 CPSH03 10078868 Ki = 10491 nM T79031 CSA7C0 10098656 IC50 = 243 nM T79031 C0LOV8 10100288 IC50 = 23 nM T79031 CK51FX 10100482 IC50 = 26 nM T79031 C9F4ER 10120976 IC50 = 2 nM T79031 CGF5W8 10121332 EC50 = 4 nM T79031 CKVH01 10121628 IC50 = 1400 nM T79031 CI3WQ9 10122378 EC50 = 12 nM T79031 CENB09 10122445 EC50 = 2 nM T79031 C8O9WX 10144519 EC50 = 6 nM T79031 CVH3A1 10145940 EC50 = 1 nM T79031 C1WOS4 10146227 IC50 = 4 nM T79031 CE46MS 10146435 IC50 = 112 nM T79031 CI4M8T 10146748 EC50 = 5 nM T79031 CSQW97 10147942 IC50 = 49 nM T79031 CO80TP 10167359 IC50 = 2800 nM T79031 C2RM3E 10167550 EC50 = 4 nM T79031 CU0BN5 10168098 EC50 = 2 nM T79031 C09NQE 10168127 IC50 = 310 nM T79031 CB6ZH0 10168228 EC50 = 4 nM T79031 CWMV50 10190314 IC50 = 4 nM T79031 CU62JC 10202734 Ki = 1600 nM T79031 C4RW7F 10211405 EC50 = 1 nM T79031 CC2I7B 10212352 IC50 = 2 nM T79031 CE7GN1 10252009 IC50 = 1700 nM T79031 CU7W8G 10253763 IC50 = 14000 nM T79031 C2UNQ0 10258545 IC50 = 126 nM T79031 CB60PQ 10258985 IC50 = 11 nM T79031 C1NJF9 10281819 EC50 = 2 nM T79031 CPA0J8 10282555 IC50 = 400 nM T79031 C4TNV3 10283187 EC50 = 0.6 nM T79031 C4S2YM 10304728 EC50 = 0.2 nM T79031 CF48GO 10305901 Ki = 8 nM T79031 CJZ98B 10324013 IC50 = 305 nM T79031 C3QN7I 10326962 IC50 = 5 nM T79031 CM46XO 10327211 IC50 = 205 nM T79031 CR21DA 10329743 IC50 = 4000000 nM T79031 CML3K5 10348155 IC50 = 43 nM T79031 CJ7N0D 10366180 IC50 = 690 nM T79031 C52CNL 10368645 IC50 = 44 nM T79031 CN89XA 10369729 IC50 = 1350 nM T79031 CQ0Y7C 10371570 IC50 = 15 nM T79031 CIA94Y 10371854 IC50 = 8 nM T79031 CZ5J7R 10391277 IC50 = 760 nM T79031 CZK1G9 10413386 IC50 = 440 nM T79031 CYL37G 10415909 IC50 = 20 nM T79031 CEYO32 10416248 IC50 = 570 nM T79031 CSW7R2 10425234 IC50 = 2400 nM T79031 C8F3EC 10438938 IC50 = 930 nM T79031 CJU80M 10439665 IC50 = 29 nM T79031 CPL7K3 10440747 Ki = 1.6 nM T79031 C9L4UD 10455044 Ki = 2900 nM T79031 CZ6GK9 10461757 IC50 = 18 nM T79031 CC9V1D 10466390 IC50 > 500000 nM T79031 CV1D8K 10468093 IC50 = 16090 nM T79031 CYE70D 10483879 IC50 = 32 nM T79031 C74JHX 10483887 IC50 = 21 nM T79031 CN68BR 10484078 IC50 = 3470 nM T79031 CF5E2S 10521609 IC50 = 333 nM T79031 C9BHN2 10533009 IC50 = 1650 nM T79031 C52YDR 10717792 IC50 > 10000 nM T79031 CXVH42 10762160 IC50 = 697 nM T79031 C30MWO 10812923 IC50 = 3300 nM T79031 CG80EQ 10908277 IC50 = 40000 nM T79031 C94QKP 10908388 Ki = 1129 nM T79031 CCBK42 10919408 IC50 = 140000 nM T79031 C1GYV7 10931081 IC50 = 353 nM T79031 CLV80Z 10974718 Ki = 10491 nM T79031 CL1S4U 10995760 IC50 = 3000 nM T79031 C03QFA 10999443 IC50 = 12560 nM T79031 C9PFL2 11013288 IC50 = 4240 nM T79031 C6F8RB 11018389 IC50 = 300 nM T79031 C9MC7V 11028241 Ki = 22423 nM T79031 CK0JO7 11050296 Ki = 3134 nM T79031 C48BLQ 11061522 Ki = 50.1 nM T79031 C5HJY1 11083054 Ki = 5.9 nM T79031 CP6Y0G 11083399 IC50 = 2000 nM T79031 CCT8U2 11093357 Ki = 5808 nM T79031 CUZ1H3 11114008 IC50 > 10000 nM T79031 CK5L8E 11125485 IC50 > 91000 nM T79031 CXS15N 11146809 Ki = 61.4 nM T79031 C3RQ9I 11157167 IC50 = 5 nM T79031 C3LJ6O 11166730 IC50 = 279 nM T79031 C6HBJ0 11168125 IC50 = 73 nM T79031 C73JDC 11169204 IC50 = 63000 nM T79031 CZ40LC 11169672 IC50 = 185 nM T79031 CEX8G1 11178891 IC50 = 91 nM T79031 CP6H3C 11180403 IC50 = 79 nM T79031 CJQM47 11183666 IC50 = 338000 nM T79031 CRXD31 11185491 IC50 = 460 nM T79031 C06BES 11192316 IC50 = 3 nM T79031 CL1OW5 11192984 IC50 = 75 nM T79031 CQ71PI 11193205 IC50 = 9560 nM T79031 CX91PV 11193493 IC50 = 17500 nM T79031 C8M7PR 11198061 IC50 > 25 nM T79031 C5ECR8 11203516 IC50 = 10 nM T79031 CXY85E 11203538 IC50 = 22000 nM T79031 C9LK4F 11204313 IC50 = 190 nM T79031 CN8IX6 11215318 IC50 = 14 nM T79031 CY7IP9 11215540 IC50 = 5 nM T79031 COWF09 11215541 IC50 = 9 nM T79031 CJHM10 11227304 IC50 = 7 nM T79031 CH81IQ 11227430 IC50 = 23 nM T79031 CH3RF8 11227663 IC50 = 25 nM T79031 C4HXV1 11232421 IC50 = 2600 nM T79031 C29MFW 11237963 Ki = 27 nM T79031 C50KSZ 11238050 IC50 = 2 nM T79031 CU0C8V 11238286 IC50 = 9 nM T79031 C0LY1A 11238352 IC50 = 40 nM T79031 CG87MJ 11250223 IC50 = 60 nM T79031 CKTJ19 11260293 IC50 > 10000 nM T79031 C0V3XN 11262463 IC50 = 4 nM T79031 C9L7RA 11262610 IC50 = 3350 nM T79031 C6PLT1 11272657 IC50 = 13 nM T79031 CB6KX3 11273691 IC50 = 117 nM T79031 CSI38B 11273865 IC50 = 7 nM T79031 CR3Z5A 11284421 IC50 = 209 nM T79031 CR3YE1 11284734 IC50 = 60 nM T79031 CU80VL 11290116 IC50 = 3700 nM T79031 C9E0FG 11295146 IC50 = 11 nM T79031 C4WK2S 11295726 IC50 = 48 nM T79031 C7FKT1 11296858 IC50 = 2 nM T79031 CNS4B0 11296859 IC50 = 2 nM T79031 C12GUA 11306629 IC50 = 20 nM T79031 CX0GT9 11307634 IC50 = 1820 nM T79031 CM3G0J 11308211 IC50 = 9 nM T79031 CY5GU3 11308212 IC50 = 5 nM T79031 CV8J9H 11308746 IC50 = 40 nM T79031 CZ7TI0 11317313 IC50 = 1100 nM T79031 CH0BE5 11318606 IC50 = 20 nM T79031 CM6Y4N 11319368 IC50 > 10000 nM T79031 CVDC34 11329962 IC50 = 144 nM T79031 C0SY2J 11330997 IC50 = 12 nM T79031 CL0P2H 11342148 IC50 = 64 nM T79031 C2LFN6 11342476 IC50 = 25 nM T79031 CR0TE8 11342515 IC50 = 2122 nM T79031 CYUS35 11342913 IC50 = 751 nM T79031 CX58CV 11354252 IC50 = 32 nM T79031 CL1D4N 11354322 IC50 = 6600 nM T79031 CT8LE6 11375895 IC50 = 350 nM T79031 C6YRP3 11376096 IC50 = 9 nM T79031 C5QL8O 11376341 IC50 = 23000 nM T79031 CY78LG 11377351 IC50 = 29 nM T79031 CI0F2X 11387554 IC50 > 100000 nM T79031 CAL5T6 11399412 IC50 = 52 nM T79031 C3RY8F 11410190 IC50 = 997 nM T79031 CHX8E5 11410816 IC50 = 10 nM T79031 CJS69P 11410845 IC50 = 720 nM T79031 CIPA26 11410903 IC50 = 14000 nM T79031 CLSW56 11413566 IC50 = 862000 nM T79031 C84MEW 11421906 IC50 = 396 nM T79031 CF86YO 11431235 IC50 = 54 nM T79031 CEU1W2 11432989 IC50 = 925 nM T79031 CNY2L9 11443660 IC50 = 8 nM T79031 CEM8Q5 11444313 IC50 = 16 nM T79031 C3ZI7O 11444912 IC50 = 48 nM T79031 CR4F1K 11456236 IC50 = 22.95 nM T79031 CLK8V9 11467715 IC50 = 8 nM T79031 C0OPF5 11467778 IC50 = 227 nM T79031 CUVZ93 11468096 IC50 = 3440 nM T79031 CH2Y7V 11478322 IC50 = 23 nM T79031 CLD65U 11479212 IC50 = 24 nM T79031 C7LAQ1 11493476 IC50 = 20300 nM T79031 CT2UK0 11495643 IC50 = 1400 nM T79031 C5QAX7 11496159 IC50 = 1000 nM T79031 CZ6X5V 11496483 IC50 = 1300 nM T79031 CW4MG8 11496999 IC50 > 5000 nM T79031 CB8RT4 11497030 IC50 = 1000 nM T79031 CRZ86I 11498384 Ki = 0.12 nM T79031 C2RXZ9 11499243 EC50 = 217000 nM T79031 CH4ZM5 11500493 IC50 = 40000 nM T79031 C4OS0M 11504350 IC50 = 110 nM T79031 C5Y9BF 11504414 IC50 = 110 nM T79031 CZN64G 11505418 IC50 = 0.89 nM T79031 C14WOL 11507920 IC50 = 9100 nM T79031 C2LD3N 11510567 IC50 = 50 nM T79031 CK0L9W 11510740 IC50 = 100 nM T79031 CUB21A 11511564 IC50 = 90 nM T79031 CH54VR 11511585 Ki = 50.12 nM T79031 CK35JZ 11512035 Ki = 3000 nM T79031 C9M3OA 11512055 IC50 = 1000 nM T79031 C7N6BE 11512310 IC50 = 4 nM T79031 CG3DO8 11512324 IC50 = 2060 nM T79031 CK70GR 11512869 Ki = 11300 nM T79031 C3P6ZU 11516577 IC50 = 40 nM T79031 CRKI87 11516654 IC50 = 1800 nM T79031 CYIV63 11517020 IC50 = 20 nM T79031 CLN34P 11517146 IC50 = 1780 nM T79031 CJCN06 11517373 IC50 = 690 nM T79031 C8R5BZ 11517807 IC50 = 1300 nM T79031 CW68BJ 11518143 IC50 > 30000 nM T79031 C5XB3T 11520033 IC50 = 5 nM T79031 CK2JD4 11525068 IC50 = 255 nM T79031 C0JGK7 11526735 IC50 = 69 nM T79031 C3M7WY 11526737 IC50 = 670 nM T79031 C1TP2W 11526803 IC50 = 5500 nM T79031 CHL65Z 11526916 IC50 = 2400 nM T79031 C2VN5E 11531131 EC50 = 680 nM T79031 C3E4UL 11531641 IC50 = 1000 nM T79031 CIK75C 11532248 IC50 = 40 nM T79031 CBP8Y9 11532527 IC50 = 850 nM T79031 CPK79W 11532880 EC50 = 90 nM T79031 C5QB4G 11533200 IC50 = 559 nM T79031 CB3O5D 11533436 IC50 = 292 nM T79031 C3M7DV 11537197 IC50 = 5600 nM T79031 C9EN6M 11537623 IC50 = 200 nM T79031 C2W8MQ 11538592 IC50 = 130 nM T79031 CT50OI 11539235 IC50 = 59.98 nM T79031 C0T2BA 11539555 IC50 = 1300 nM T79031 C6CVW2 11539562 EC50 = 20 nM T79031 CR93VK 11539712 IC50 = 34 nM T79031 C6FED7 11541583 IC50 = 21 nM T79031 C2IL9N 11543843 EC50 = 16000 nM T79031 CS8MV6 11544960 EC50 = 5100 nM T79031 CPO30U 11544998 Ki = 290 nM T79031 C0KY4O 11545958 IC50 = 36 nM T79031 C4IP5W 11546946 IC50 = 980 nM T79031 CHT39Z 11549051 Ki = 71 nM T79031 CLWN51 11550876 IC50 = 38000 nM T79031 CYEL51 11553053 EC50 = 4600 nM T79031 C1EF0M 11553329 IC50 = 1300 nM T79031 CSL71C 11553983 IC50 = 119.95 nM T79031 CZJ64S 11555685 IC50 = 46 nM T79031 CE9ZI8 11556254 IC50 = 5 nM T79031 CWR28P 11556734 IC50 = 3 nM T79031 CZ07VP 11560610 IC50 = 630 nM T79031 C8CA9X 11561538 IC50 = 100 nM T79031 CL92RI 11562095 IC50 = 1600 nM T79031 CZ23YB 11565240 IC50 = 16000 nM T79031 CQ0Y1L 11565289 IC50 = 79000 nM T79031 C5Y2ZJ 11566309 Ki = 59 nM T79031 C5N8OY 11567707 IC50 = 1200 nM T79031 CNJX56 11569561 IC50 = 35 nM T79031 CO0AV9 11569760 IC50 = 1700 nM T79031 COP47N 11573395 IC50 = 5200 nM T79031 C5RNW0 11574638 IC50 = 2450 nM T79031 CTN4X2 11575549 IC50 > 10000 nM T79031 C86SBR 11575810 IC50 = 1500 nM T79031 CS2WU3 11576068 IC50 = 590 nM T79031 C8OUD5 11576737 IC50 = 276 nM T79031 C5UR7S 11578047 IC50 = 0.7 nM T79031 CBQ68E 11578322 IC50 = 1.4 nM T79031 CR8AL4 11582999 Ki = 39 nM T79031 CE6CH3 11583947 IC50 = 160 nM T79031 CC8T2P 11584133 IC50 = 1250 nM T79031 C4WYG7 11587584 IC50 = 190000 nM T79031 CA29QF 11589453 IC50 = 89.95 nM T79031 CYO9W4 11589920 IC50 = 3000 nM T79031 C9FI7P 11590166 IC50 = 437 nM T79031 C89CMR 11592145 IC50 = 7 nM T79031 CJ4OB9 11594328 IC50 = 27000 nM T79031 CA2Q5C 11594966 IC50 = 380 nM T79031 C1A7SE 11596660 IC50 = 590 nM T79031 CD6KY0 11596715 IC50 > 20000 nM T79031 CUP02D 11596983 IC50 = 3400 nM T79031 CW79HO 11598623 IC50 = 1200 nM T79031 CT2HP4 11598634 IC50 = 25000 nM T79031 C0EOP4 11604171 IC50 = 680 nM T79031 CV30CG 11604834 IC50 = 536 nM T79031 CXQ2P7 11605160 IC50 = 1800 nM T79031 CZ1V8Y 11606008 IC50 = 600 nM T79031 C12SFR 11606910 IC50 = 4 nM T79031 CAP4I0 11608786 IC50 = 25000 nM T79031 C92XGC 11609507 Ki = 160 nM T79031 CT97EJ 11611402 IC50 = 50 nM T79031 CL9V5H 11611694 IC50 = 310 nM T79031 CA2L6B 11613176 IC50 = 79 nM T79031 C68NYG 11613697 IC50 = 1830 nM T79031 CAGB98 11613886 IC50 = 29900 nM T79031 C1PSL5 11614083 IC50 = 3 nM T79031 CFU9Q3 11618427 EC50 = 5100 nM T79031 CMW5Y1 11618935 IC50 = 942 nM T79031 CMQ38D 11619220 IC50 = 550 nM T79031 CAP36L 11619283 IC50 = 255 nM T79031 CQ7A5C 11620172 IC50 = 68 nM T79031 C7ZWK0 11620576 IC50 = 220 nM T79031 C9HXM0 11621130 IC50 = 5000 nM T79031 CLI21W 11621627 Ki = 33 nM T79031 CV29MK 11621744 IC50 = 2.5 nM T79031 C1Y5SJ 11621924 IC50 = 2.7 nM T79031 CI0BT7 11623676 IC50 = 6500 nM T79031 C9R6UV 11624078 Ki = 130 nM T79031 CJ13UK 11626083 IC50 = 1400 nM T79031 CH12YA 11628169 IC50 = 4740 nM T79031 C7P1VQ 11628699 IC50 = 6.5 nM T79031 C0TQM3 11628951 IC50 = 5 nM T79031 CVP4Z0 11630139 IC50 = 34000 nM T79031 CO7L8Z 11631207 Ki = 57 nM T79031 CUD76B 11632510 EC50 = 420 nM T79031 C78KYL 11633041 EC50 = 1630 nM T79031 C2BY3T 11633167 IC50 = 4200 nM T79031 CC74NS 11633817 IC50 = 110 nM T79031 C2QC4B 11633904 IC50 = 70 nM T79031 CH6JI3 11634931 IC50 = 151 nM T79031 C7IH1Z 11638363 IC50 = 1600 nM T79031 COC2F0 11639859 IC50 = 149.97 nM T79031 CED2Y7 11640634 IC50 = 239 nM T79031 CBI2Q1 11642048 IC50 = 40 nM T79031 CNT76I 11642873 IC50 = 5.7 nM T79031 C46FQR 11643019 IC50 = 2 nM T79031 CX37JT 11645215 IC50 = 19800 nM T79031 CY1C4O 11646236 IC50 = 1600 nM T79031 C8BX9Z 11647679 IC50 = 1650 nM T79031 C8DZG9 11647909 IC50 = 210 nM T79031 C7M0KO 11647968 IC50 = 1100 nM T79031 C6MH7K 11648455 IC50 = 60 nM T79031 CR16HF 11649408 Ki = 1300 nM T79031 C1JAC8 11650016 IC50 = 6 nM T79031 CH5J1Y 11650532 IC50 = 2.1 nM T79031 CH2GE3 11652923 IC50 = 5900 nM T79031 C0UXN3 11654224 EC50 = 860 nM T79031 CSKL32 11654876 EC50 = 680 nM T79031 CT13BA 11655737 IC50 = 370 nM T79031 CEU6R3 11655813 IC50 = 665 nM T79031 CMT32N 11655970 IC50 = 1300 nM T79031 CF7LR8 11656491 IC50 = 1400 nM T79031 C7FL0K 11657376 Ki = 120 nM T79031 C2OKH7 11659487 IC50 = 25000 nM T79031 CJP6A2 11662513 Ki = 15848.93 nM T79031 C9ZOM3 11663095 IC50 = 150 nM T79031 CW9MD3 11664318 IC50 = 4 nM T79031 C1UQ7K 11664850 IC50 = 48 nM T79031 C03OWT 11666379 IC50 = 3500 nM T79031 C4PXM5 11668120 EC50 = 370 nM T79031 C14JYI 11668187 IC50 = 30 nM T79031 CUD4R5 11669598 IC50 = 90 nM T79031 CL54AU 11669760 IC50 = 10000 nM T79031 C59UWB 11673750 IC50 = 120000 nM T79031 C4FN0W 11675187 IC50 = 1700 nM T79031 C8SXN1 11676068 IC50 = 1150 nM T79031 CEI62A 11676832 IC50 = 79 nM T79031 C2HBA9 11677867 IC50 = 87 nM T79031 C80VBO 11679203 IC50 = 2.6 nM T79031 CIQL54 11679286 IC50 = 10 nM T79031 CM19TA 11681539 IC50 = 24000 nM T79031 CY47BE 11683112 IC50 = 1430 nM T79031 C4G6YQ 11684817 IC50 = 170 nM T79031 CZ07AQ 11689885 IC50 = 900 nM T79031 C6H8TK 11691007 IC50 = 410 nM T79031 C7SPG0 11692473 IC50 = 12 nM T79031 CB2GA5 11697219 IC50 = 3000 nM T79031 CGC2T9 11698483 IC50 = 1200 nM T79031 C0AR2C 11698518 IC50 = 630 nM T79031 CBP7Q2 11699253 IC50 = 760 nM T79031 C3XA6V 11699481 IC50 = 580 nM T79031 CR02ZX 11699482 IC50 = 580 nM T79031 C4T8XV 11700105 IC50 = 100 nM T79031 C8ZE7W 11700321 Ki = 1 nM T79031 CV6CD0 11702315 IC50 = 32000 nM T79031 CO8V5F 11705058 IC50 = 1900 nM T79031 CS89KD 11705108 EC50 = 2560 nM T79031 C2IW8S 11705141 IC50 = 460 nM T79031 CQ58VW 11707063 IC50 = 120 nM T79031 CK73DU 11710655 EC50 = 5100 nM T79031 C9ZC7H 11710986 IC50 = 2250 nM T79031 CBJ08S 11711024 EC50 = 1400 nM T79031 C3ZUI4 11714054 IC50 = 7 nM T79031 C7ZRM9 11719190 IC50 = 420 nM T79031 C0G5SJ 11719407 IC50 = 410 nM T79031 C6EQ2H 11719839 IC50 = 283 nM T79031 CYG3Q1 11720331 IC50 = 2 nM T79031 CVHG04 11720625 IC50 = 10000 nM T79031 CJ4N5Y 11738522 Ki = 720 nM T79031 CB46YU 11753622 IC50 = 5 nM T79031 CHEI17 11754571 IC50 = 47 nM T79031 CGE50S 11757267 Ki = 1700 nM T79031 CF1CZ0 11765081 IC50 = 20 nM T79031 CN7AX1 11765192 IC50 = 13 nM T79031 CJN0K9 11765311 IC50 = 210 nM T79031 C2S4IA 11765692 IC50 = 21 nM T79031 CW1SG6 11768241 IC50 = 46 nM T79031 C8LJ4X 11776869 IC50 = 8220 nM T79031 CPX94C 11785473 IC50 = 11 nM T79031 CF1RT6 11785879 IC50 = 48.9 nM T79031 CG2HY0 11785880 IC50 = 15 nM T79031 CVQ7O2 11786748 IC50 = 15 nM T79031 CAT4Q9 11787283 IC50 = 139 nM T79031 CL81HQ 11819216 IC50 = 300 nM T79031 CR5M7I 11845063 IC50 > 10000 nM T79031 CV8XS9 11845069 IC50 > 10000 nM T79031 CEK56D 11845403 IC50 > 10000 nM T79031 C8H1ES 11845584 IC50 > 10000 nM T79031 C0W1KA 11845953 IC50 > 10000 nM T79031 CJ34FE 11845955 IC50 > 10000 nM T79031 CX34FU 11846304 IC50 = 20000 nM T79031 CUON19 11846305 IC50 = 16900 nM T79031 CI72TF 11846306 IC50 > 10000 nM T79031 C38JYH 11846473 IC50 = 9000 nM T79031 CICT21 11846474 IC50 > 10000 nM T79031 C8YEH5 11846475 IC50 > 10000 nM T79031 CKR6T3 11846476 IC50 > 10000 nM T79031 CHC79W 11846478 IC50 > 10000 nM T79031 CPO8E1 11846645 IC50 = 1970 nM T79031 CG1UP6 11846815 IC50 > 10000 nM T79031 CE2OQ9 11846965 IC50 > 10000 nM T79031 CR3G5X 11846966 IC50 = 1300 nM T79031 C25PFL 11846967 IC50 > 10000 nM T79031 CU2TQ6 11846968 IC50 > 10000 nM T79031 CVQ9U5 11847590 IC50 = 12000 nM T79031 CP93HT 11962092 IC50 = 4.8 nM T79031 C5S2IK 11962093 IC50 = 1.2 nM T79031 CLP92O 11963435 IC50 > 30000 nM T79031 C3KL1E 11966417 IC50 = 50000 nM T79031 CS82QV 11967065 Ki = 8 nM T79031 C5L8QT 11983210 Ki = 20 nM T79031 CGOD35 11990754 IC50 = 20 nM T79031 CQ8SJ5 11990755 IC50 = 40 nM T79031 CIKT23 11995758 IC50 = 1890 nM T79031 CF9NQ6 11995759 IC50 = 680 nM T79031 CYF60T 11995761 IC50 = 590 nM T79031 CC8W5S 11995764 IC50 = 8300 nM T79031 C0O2KV 11995892 IC50 = 630 nM T79031 CRT1N8 11997830 IC50 = 930 nM T79031 CP40AD 11997831 IC50 = 200 nM T79031 C4TOJ6 11997832 IC50 = 6900 nM T79031 C0P6SQ 11997981 IC50 = 260 nM T79031 C4RGE9 11997983 IC50 = 750 nM T79031 CA97TM 12120708 IC50 = 600 nM T79031 CJC3N0 12146686 IC50 = 17000 nM T79031 CTOG21 12402626 IC50 = 41200 nM T79031 C4G1PQ 12507854 IC50 = 20010 nM T79031 CL2KU0 13070818 IC50 > 2000000 nM T79031 C5FCE3 14018347 IC50 > 3000000 nM T79031 C2T8ZO 14977406 IC50 = 13410 nM T79031 CH4BX8 15081178 IC50 = 4770 nM T79031 CKD36Y 15940224 IC50 = 4 nM T79031 C4F9TQ 15941301 Ki = 3900 nM T79031 CJH9P6 15941302 Ki = 670 nM T79031 C7F3BW 15941303 Ki = 2800 nM T79031 CV4UH9 15941304 Ki = 290 nM T79031 C79YMT 15941305 Ki = 870 nM T79031 C2PSD7 15941443 Ki = 4000 nM T79031 CG3ZY1 15941444 Ki = 210 nM T79031 CW2ZY9 15941577 Ki = 480 nM T79031 CLU58A 15941580 Ki = 120 nM T79031 CO7YL9 15947487 Ki = 26 nM T79031 C1FQ3D 15949752 IC50 = 93 nM T79031 CR4G6J 15949919 IC50 = 60 nM T79031 CQ3GX2 15950003 EC50 = 140 nM T79031 C3CI9Z 15950004 IC50 = 10 nM T79031 C2BQ4V 15950005 IC50 = 30 nM T79031 C6QD9U 15950006 EC50 = 700 nM T79031 CW4US1 15950085 EC50 = 900 nM T79031 CZM1C9 15950086 IC50 = 30 nM T79031 C8Y6UT 15950518 IC50 = 240 nM T79031 CAPV27 15950520 IC50 = 630 nM T79031 C20LCO 15950595 IC50 = 100 nM T79031 C6DCB3 15950597 IC50 = 29.99 nM T79031 C49WLN 15950662 IC50 = 139.96 nM T79031 CK4L8W 15950666 IC50 = 60 nM T79031 C0OCS6 15950667 IC50 = 79.98 nM T79031 C3WIC9 15951413 IC50 = 2679.17 nM T79031 C0J9PD 15951416 IC50 = 130 nM T79031 CSQ3X1 15951420 IC50 = 50 nM T79031 C8IZR0 15951484 IC50 = 59.98 nM T79031 CB1G7D 15951486 IC50 = 250 nM T79031 CNPJ39 15951487 IC50 = 39.99 nM T79031 C2XJU6 15951488 IC50 = 69.98 nM T79031 CE67NK 15951489 IC50 = 29.99 nM T79031 CW6S0H 15981486 IC50 = 2 nM T79031 CYW5P8 15988250 IC50 = 100000 nM T79031 C85PQC 15993676 IC50 = 100000 nM T79031 CQ93FI 15995071 IC50 = 100000 nM T79031 C8KLU4 15999741 IC50 = 100000 nM T79031 C16ATP 16000372 IC50 = 100000 nM T79031 CION47 16003623 IC50 = 100000 nM T79031 C6A7LF 16004116 IC50 = 100000 nM T79031 CGY5P4 16004117 IC50 = 100000 nM T79031 CS8EY3 16038399 IC50 = 90 nM T79031 C5HUB3 16040323 IC50 = 80 nM T79031 CJ1H2F 16043232 IC50 = 5.6 nM T79031 C0QAD8 16050550 EC50 = 44 nM T79031 C1CEU6 16050551 IC50 = 330 nM T79031 CX8O6Q 16050552 EC50 = 570 nM T79031 CYQ7X3 16050553 EC50 = 760 nM T79031 C2WR8B 16050640 EC50 = 930 nM T79031 CF5EC0 16050641 EC50 = 190 nM T79031 CN0F8Z 16050834 IC50 = 1080 nM T79031 CD5W4A 16050837 IC50 = 4797.33 nM T79031 C4DO8C 16050931 IC50 = 990 nM T79031 C8R6HZ 16050932 IC50 = 1039.92 nM T79031 C21JUT 16050937 IC50 = 390 nM T79031 C72ZAL 16050938 IC50 = 950.6 nM T79031 CL35CA 16051038 IC50 = 1240 nM T79031 C2CJ4S 16051040 IC50 = 1390 nM T79031 CQCJ80 16051495 IC50 = 1360 nM T79031 CRAS90 16051584 IC50 = 7860 nM T79031 C0Q2MC 16051586 IC50 = 40 nM T79031 CW6CX4 16051696 IC50 = 860 nM T79031 CL4I9N 16051697 IC50 = 210 nM T79031 CE3L1D 16051698 IC50 = 100 nM T79031 C1KRO6 16061967 IC50 = 2 nM T79031 C4MX6F 16062196 IC50 = 10 nM T79031 CAI1G0 16062314 IC50 = 17 nM T79031 CAY1B5 16090342 IC50 = 600 nM T79031 CP5G7V 16090348 IC50 = 110 nM T79031 C2CK4A 16092132 Ki = 20 nM T79031 COPC57 16094305 IC50 = 200 nM T79031 C6FGY9 16094306 IC50 = 1370 nM T79031 CF0Q8I 16094307 IC50 = 138 nM T79031 C6Y8MP 16094311 IC50 = 12500 nM T79031 C0QGD1 16094312 IC50 = 2700 nM T79031 CWGX63 16094313 IC50 = 27 nM T79031 C2WM0N 16109345 IC50 = 130 nM T79031 C7MV4N 16109346 IC50 = 70 nM T79031 CKC8Z5 16109350 IC50 = 500 nM T79031 CT1F3Y 16109351 IC50 = 200 nM T79031 CXC0E3 16109352 IC50 = 130 nM T79031 C2HMT5 16113206 IC50 = 10 nM T79031 CX39UL 16113753 EC50 = 160 nM T79031 C81OJE 16113965 IC50 = 30 nM T79031 CJDF09 16129583 IC50 = 11 nM T79031 CC64JE 16148440 IC50 = 410 nM T79031 C4E6OY 16148496 IC50 = 40000 nM T79031 CH1B3X 16148708 IC50 > 200000 nM T79031 C4L0VN 16149641 IC50 = 500 nM T79031 C5Z1RK 16149643 IC50 = 30 nM T79031 CZX90D 16149773 IC50 > 200000 nM T79031 CL26VD 16659019 Ki = 1.8 nM T79031 CU62LO 16659020 Ki = 136 nM T79031 CK9G4O 16659021 Ki = 315 nM T79031 CGU76F 16659022 Ki = 27 nM T79031 CJ16IR 16659063 Ki = 788 nM T79031 C73FHN 16659067 Ki = 52.5 nM T79031 C01GFZ 16659107 Ki = 438 nM T79031 C1KY6O 16722358 IC50 = 150000 nM T79031 CVM2G8 16725331 IC50 = 13 nM T79031 C1XN0F 16725801 IC50 = 77 nM T79031 CZ2DN8 16725908 IC50 = 6 nM T79031 CEAK02 16726085 IC50 = 30 nM T79031 CRW5Q2 16730753 IC50 = 12 nM T79031 CK6CL9 16741238 Ki = 900 nM T79031 CI7Z6F 16741239 Ki = 8 nM T79031 CKHB98 16741878 IC50 = 19540 nM T79031 C2K9NL 16748452 IC50 = 173 nM T79031 C82CQR 16750202 IC50 > 10000 nM T79031 CH9Y5B 17159064 IC50 = 3000 nM T79031 C5ZMI9 17159212 IC50 = 5300 nM T79031 CF6ZW1 17159244 IC50 = 13000 nM T79031 C80YMT 17159252 IC50 = 430 nM T79031 CF0N8R 17749735 Ki = 270 nM T79031 C42ZVI 17756380 Ki = 158 nM T79031 CMXW48 21085652 IC50 = 30 nM T79031 CU2E5X 21087080 IC50 = 4131 nM T79031 C2FBA3 21672659 IC50 > 10000 nM T79031 CW3AO5 21826766 IC50 > 500000 nM T79031 C7OEP8 22331258 IC50 = 100000 nM T79031 C1I0HR 22427309 IC50 = 100000 nM T79031 CX4H0M 22674193 IC50 = 400000 nM T79031 CMXJ30 23625795 IC50 > 10000 nM T79031 C2JXU0 23644687 IC50 = 82 nM T79031 C89VMI 23644698 Ki = 217.6 nM T79031 CRVN47 23644701 IC50 = 8 nM T79031 C3VQK5 23644703 IC50 = 418 nM T79031 C1LIH9 23644704 IC50 = 1400 nM T79031 CR1DT2 23644705 IC50 = 115 nM T79031 C3JWR0 23644706 IC50 = 110 nM T79031 CN7DC2 23644707 IC50 = 115 nM T79031 CR7K1W 23644708 IC50 = 348 nM T79031 CXJ41P 23646327 IC50 = 9704 nM T79031 C0IGT6 23646330 IC50 = 285 nM T79031 CCKB26 23646331 IC50 = 4925 nM T79031 CCU65J 23646332 IC50 = 260 nM T79031 C4WTR7 23647188 IC50 = 2397 nM T79031 C8DJ0O 23647273 IC50 = 980 nM T79031 C50XEQ 23647274 IC50 = 1500 nM T79031 CQ0Y1I 23647275 IC50 = 1400 nM T79031 CISN90 23647276 IC50 = 5500 nM T79031 C8ON7P 23647277 IC50 = 5900 nM T79031 C0FH3Q 23647278 IC50 = 1300 nM T79031 CTN78W 23647279 IC50 = 4630 nM T79031 CWR50S 23647280 IC50 = 450 nM T79031 C7QC4Y 23647281 IC50 = 240 nM T79031 C8JXG2 23647282 IC50 = 180 nM T79031 C1U6EJ 23647283 IC50 = 730 nM T79031 C54ZEQ 23647284 IC50 = 420 nM T79031 CKZ2T9 23647285 IC50 = 21000 nM T79031 CZP52T 23647286 IC50 = 3400 nM T79031 CP4S6K 23647287 IC50 = 100000 nM T79031 CJVE50 23647289 Ki = 87.2 nM T79031 C7FA0O 23647290 Ki = 61.4 nM T79031 CHL32N 23647291 Ki = 28.4 nM T79031 C4G2TH 23647292 Ki = 108.2 nM T79031 C96CZH 23647293 Ki = 112.1 nM T79031 C0T8KQ 23647294 IC50 > 10000 nM T79031 C17VPL 23647295 IC50 = 120 nM T79031 CG46BK 23647296 IC50 = 100 nM T79031 CMY6Q4 23647310 IC50 > 10000 nM T79031 C8IY5K 23647384 IC50 = 74 nM T79031 CVQ0Y4 23647390 IC50 = 31 nM T79031 CAJN03 23647391 IC50 = 39 nM T79031 CZQ5A9 23647392 IC50 = 67 nM T79031 CX8ME3 23647393 IC50 = 24 nM T79031 CR6BI7 23647394 IC50 = 24 nM T79031 C5Z1FD 23647395 IC50 = 462 nM T79031 CWMS83 23647396 IC50 = 5900 nM T79031 C53ZIT 23647400 IC50 = 9900 nM T79031 C4XFA0 23647401 IC50 = 223 nM T79031 CMT72O 23647402 IC50 = 674 nM T79031 C1WZS4 23647403 IC50 = 317 nM T79031 CZ0XL6 23647406 IC50 > 10000 nM T79031 CHJC53 23647407 IC50 > 100000 nM T79031 CWM6S0 23647408 IC50 = 2900 nM T79031 C15KHL 23647409 IC50 = 5400 nM T79031 CG79IQ 23647410 IC50 = 1100 nM T79031 CYPK85 23647411 IC50 = 90 nM T79031 CNZ90K 23647412 IC50 = 300 nM T79031 CK40YS 23657802 IC50 = 33 nM T79031 C4BR2E 23657804 IC50 = 1800 nM T79031 C5WBN8 23661698 IC50 = 1700 nM T79031 CVL23N 23730798 IC50 = 160 nM T79031 CU57QT 23730803 IC50 = 480000 nM T79031 C9GEC0 23730921 IC50 = 140000 nM T79031 C4P7UO 23731036 IC50 = 3800 nM T79031 C7MW0V 23731038 IC50 = 35000 nM T79031 C8J3DH 23769141 IC50 = 100000 nM T79031 CAVW67 24280127 IC50 = 500000 nM T79031 CZFK29 24280444 IC50 = 500000 nM T79031 CBV08C 24280464 IC50 = 500000 nM T79031 C92YOQ 24289443 IC50 = 400000 nM T79031 CQ6MC2 24745770 Ki = 5 nM T79031 CG3M9A 24745771 Ki = 5 nM T79031 CFT94C 24764598 Ki = 5 nM T79031 C1XWQ9 24772565 Ki = 210 nM T79031 CI27XV 24772624 Ki = 110 nM T79031 CZRE74 24772625 Ki = 140 nM T79031 CY4VD2 24772627 Ki = 78 nM T79031 CKTR40 24772696 Ki = 100 nM T79031 CEI3N7 24794397 IC50 = 3 nM T79031 C2VT1S 24801864 Ki = 449 nM T79031 CT96WK 24801865 Ki = 5001 nM T79031 C7BK3P 24808496 IC50 = 14 nM T79031 CJUX10 24808497 Ki = 3 nM T79031 CY0TD7 24871744 IC50 = 107.15 nM T79031 C6FPQ4 24873157 IC50 = 100 nM T79031 CS13TR 24873277 IC50 = 28.84 nM T79031 CIX89B 24873279 IC50 = 40.74 nM T79031 C06DKB 24875236 IC50 = 90.3 nM T79031 CE05DA 24877512 IC50 = 190 nM T79031 CB9DT6 24877514 IC50 = 150 nM T79031 C3EHC6 24877515 IC50 = 990 nM T79031 C1ILH2 24877517 IC50 = 2800 nM T79031 CV7FB1 24877625 IC50 = 1500 nM T79031 C8AJ1S 24877631 IC50 = 950 nM T79031 CA37MN 24877744 IC50 = 1800 nM T79031 C4SZA8 24877746 IC50 = 1100 nM T79031 CUW1D7 24877749 IC50 = 760 nM T79031 CFJ87K 24877750 IC50 = 2300 nM T79031 C9IKJ2 24877858 IC50 = 370 nM T79031 CWM1Q4 24878892 IC50 = 101.38 nM T79031 CTO0H5 24878893 IC50 = 120 nM T79031 CKWX57 24878894 IC50 = 62.94 nM T79031 CF0Q3S 24878945 IC50 = 120 nM T79031 C09LYN 24878946 IC50 = 120 nM T79031 CI54AT 24878947 IC50 = 140 nM T79031 CU29JQ 24882306 IC50 = 0.4 nM T79031 C8LQ5C 24882338 IC50 = 13 nM T79031 CMJK34 24882477 IC50 = 14 nM T79031 CG0Z5M 24883482 IC50 > 250000 nM T79031 CY08DL 24883483 IC50 > 250000 nM T79031 CLW51O 24936061 IC50 = 99 nM T79031 C32SYP 24950594 EC50 = 200 nM T79031 C6WD3C 24969880 IC50 = 1000 nM T79031 CR8YI5 24989869 IC50 = 89.13 nM T79031 C5VK7J 24997367 IC50 = 1000 nM T79031 CQ6NH9 24997666 IC50 = 720 nM T79031 CEY73X 24997667 IC50 = 8.6 nM T79031 C4LF6D 24997668 IC50 = 4 nM T79031 CM9U5L 25008440 IC50 = 14 nM T79031 C1PR9E 25008964 IC50 = 50 nM T79031 C4P9OL 25013704 IC50 = 263.03 nM T79031 C6UCX2 25063358 Ki = 3300 nM T79031 COY78F 25063486 Ki = 460 nM T79031 CA54VF 25063645 IC50 > 10000 nM T79031 C42POG 25063685 Ki = 3800 nM T79031 CT9MX8 25066444 Ki = 2 nM T79031 CO7MQ2 25069561 EC50 = 30 nM T79031 C8ANG7 25070193 EC50 = 90 nM T79031 C0T8LP 25070195 EC50 = 150 nM T79031 CM37LQ 25072736 IC50 = 15 nM T79031 CDY56W 25072741 EC50 = 30 nM T79031 C0UO6V 25073049 IC50 = 30 nM T79031 CL3QK6 25096211 IC50 = 3.1 nM T79031 C2UWA1 25096462 IC50 = 30 nM T79031 CZV97Q 25096707 IC50 = 340 nM T79031 C3H6BD 25110732 IC50 = 12 nM T79031 C93HLR 25113163 IC50 = 37 nM T79031 CMYC57 25115954 IC50 = 0.93 nM T79031 C4E9MK 25120557 IC50 = 1710 nM T79031 CU7P0M 25120899 IC50 = 565 nM T79031 C4KM6T 25121609 IC50 = 744 nM T79031 CXO60C 25127299 IC50 = 41 nM T79031 CNTF43 25127621 EC50 = 100 nM T79031 C4E0MJ 25127622 IC50 = 20 nM T79031 C21DIX 25138203 IC50 = 24000 nM T79031 C1AY4Q 25138204 IC50 = 16000 nM T79031 CC5M6R 25138205 IC50 = 30000 nM T79031 CA78FI 25138206 IC50 = 110000 nM T79031 CHEJ69 25138207 IC50 = 69000 nM T79031 C8LK9F 25138208 IC50 > 600000 nM T79031 C5QDG2 25138209 IC50 = 570000 nM T79031 C0L3CZ 25138210 IC50 > 600000 nM T79031 C7DAF9 25138211 IC50 > 600000 nM T79031 C2QG9U 25138212 IC50 > 600000 nM T79031 CDF6M3 25138213 IC50 > 1600000 nM T79031 CCF76H 25138214 IC50 = 317000 nM T79031 CT52IW 25138215 IC50 = 15000 nM T79031 C5OX0H 25138216 IC50 = 219000 nM T79031 C9A6QG 25138217 IC50 = 19000 nM T79031 CDNA34 25138218 IC50 = 37000 nM T79031 CXN7P5 25138219 IC50 = 21000 nM T79031 CQZ97A 25142134 IC50 = 7.3 nM T79031 C6S8AH 25142266 IC50 = 20.4 nM T79031 C4J5ET 25143473 IC50 = 1.9 nM T79031 CWF5Z3 25143506 IC50 > 30000 nM T79031 CLAI84 25147572 IC50 = 18330 nM T79031 C3O5UD 25154200 IC50 = 200 nM T79031 CEUT61 25156748 Ki = 3 nM T79031 C9WN6Q 25156749 Ki = 3.3 nM T79031 CG54TK 25157024 Ki = 3.1 nM T79031 CH8YV1 25157025 Ki = 2.1 nM T79031 COK8S4 25163980 IC50 = 1400 nM T79031 C6YWX8 25163981 IC50 = 590 nM T79031 CKM2U5 25163982 IC50 = 27 nM T79031 CBH2U0 25166287 IC50 = 96 nM T79031 C42BVF 25166288 IC50 = 140 nM T79031 CL8B0V 25166485 IC50 = 360 nM T79031 CP89ZX 25181420 IC50 = 63 nM T79031 C4JQ0L 25181421 IC50 = 56 nM T79031 C3XDW1 25184934 EC50 = 900 nM T79031 CS2MU5 25184935 EC50 = 1500 nM T79031 CXE56W 25184936 EC50 = 300 nM T79031 CF91ST 25184937 IC50 = 80 nM T79031 CSM9C5 25190481 IC50 = 380 nM T79031 CU80RW 25190482 IC50 = 250 nM T79031 CK48PJ 25190483 IC50 = 280 nM T79031 CW6QJ1 25190484 IC50 = 160 nM T79031 CKZ2Q7 25190485 IC50 = 50 nM T79031 CWN51E 25190486 IC50 = 21 nM T79031 C69RHT 25190487 IC50 = 5 nM T79031 CT8N2P 25190488 IC50 = 11 nM T79031 CJ6SA2 25190489 IC50 = 5 nM T79031 CESB62 25190490 IC50 = 34 nM T79031 CLS3O2 25190491 IC50 = 34 nM T79031 CZY6C4 25190492 IC50 = 18 nM T79031 C04QGB 25190493 IC50 = 12 nM T79031 CF8U0N 25190494 IC50 = 8 nM T79031 CX4PB5 25190495 IC50 = 26 nM T79031 CKYP06 25190496 IC50 = 40 nM T79031 CNXG37 25190497 IC50 = 2690 nM T79031 CTS92Q 25190499 IC50 = 12 nM T79031 CY02QR 25190500 IC50 = 12 nM T79031 CYN2X5 25195985 IC50 = 28 nM T79031 CZP06K 25195988 IC50 = 56 nM T79031 COZ9A0 25196089 IC50 = 11 nM T79031 CGWR85 25196090 IC50 = 6 nM T79031 CU8ON3 25232084 Ki = 284 nM T79031 C60XDJ 25232085 Ki = 19004 nM T79031 C40ITP 25232817 Ki = 260 nM T79031 CA9K0S 25232818 Ki = 4957 nM T79031 C5G2BP 25232984 Ki = 51 nM T79031 CR9O7I 25232986 Ki = 3514 nM T79031 CSO74W 25233156 Ki = 267 nM T79031 CI68AZ 25233160 Ki = 6768 nM T79031 C6E5PM 25233329 Ki = 818 nM T79031 C9JEA2 25233330 Ki = 272 nM T79031 CFY28W 25233331 Ki = 867 nM T79031 C9XA8E 25233503 Ki = 53 nM T79031 C6CAS8 25233845 Ki = 3500 nM T79031 CMS9A5 25233846 Ki = 8177 nM T79031 C8TF6A 33746207 IC50 = 562000 nM T79031 CMV27B 42636931 IC50 = 150 nM T79031 CQH0F2 42636932 IC50 = 2 nM T79031 CIFH60 42643933 IC50 = 4000 nM T79031 CP3LE8 42644642 IC50 = 19000 nM T79031 C2K9JH 42646800 IC50 = 47000 nM T79031 C1E5GI 43824597 IC50 = 2600 nM T79031 COI2D4 44123817 IC50 = 98.7 nM T79031 C25ELB 44143088 IC50 = 63095.73 nM T79031 CJ5CG9 44143249 IC50 = 3700 nM T79031 CN7WQ5 44143250 IC50 = 2400 nM T79031 CV5SI1 44143251 IC50 = 1600 nM T79031 C85TLI 44143252 IC50 = 7600 nM T79031 C3RO7F 44143253 IC50 = 250 nM T79031 C6SEQ5 44143255 IC50 = 2100 nM T79031 CJL9X6 44143256 IC50 = 2500 nM T79031 C6QY9W 44143257 IC50 = 40 nM T79031 CXV1A7 44143258 IC50 = 63 nM T79031 CWI68J 44143259 IC50 = 110 nM T79031 CNQ97G 44143260 IC50 = 23 nM T79031 C95LPG 44143261 IC50 = 18 nM T79031 CV9K7F 44143262 IC50 = 19 nM T79031 C0WRT2 44143263 IC50 = 23 nM T79031 CWQ6L4 44143264 IC50 = 26 nM T79031 CZ9MQ7 44143265 IC50 = 28 nM T79031 C8EI0C 44143266 IC50 = 34 nM T79031 CAJ0I2 44143267 IC50 = 40 nM T79031 C7AH8B 44143268 IC50 = 87 nM T79031 CFJ82W 44143269 IC50 = 210 nM T79031 CQ34LK 44143270 IC50 = 420 nM T79031 C7FQ8W 44143271 IC50 = 6 nM T79031 CCUX36 44143272 IC50 = 40 nM T79031 CDR56H 44143274 IC50 = 19 nM T79031 CNWC13 44143275 IC50 = 91 nM T79031 C4C0WD 44143276 IC50 = 190 nM T79031 C5SLK9 44143277 IC50 = 8 nM T79031 C39WZR 44143278 IC50 = 26 nM T79031 CVF5L8 44143280 IC50 = 1574 nM T79031 CPX9B2 44143282 IC50 = 20 nM T79031 C6CQM2 44143283 IC50 = 8 nM T79031 CDEU24 44143285 IC50 = 360 nM T79031 CD8WS6 44143286 IC50 = 250 nM T79031 CK62TO 44189143 IC50 = 1 nM T79031 C7ZNM2 44193108 IC50 = 18000 nM T79031 C9D1YN 44193111 IC50 = 12000 nM T79031 CQ90YP 44193304 IC50 = 2850 nM T79031 C23BVR 44197099 IC50 < 1000 nM T79031 CB48HS 44197116 IC50 < 1000 nM T79031 CR0BI1 44197118 IC50 < 1000 nM T79031 C5AW6R 44197119 IC50 < 1000 nM T79031 C6HF1B 44197136 IC50 < 1000 nM T79031 CN4A9C 44197137 IC50 < 1000 nM T79031 CDC8A1 44197138 IC50 < 1000 nM T79031 C7VO3S 44197139 IC50 < 1000 nM T79031 CVW8R0 44197162 IC50 < 1000 nM T79031 CPA52Y 44197163 IC50 < 1000 nM T79031 CG4QP1 44197191 IC50 < 1000 nM T79031 CJ05UB 44197192 IC50 < 1000 nM T79031 CQFO09 44197193 IC50 < 1000 nM T79031 CQ02XS 44197219 IC50 < 1000 nM T79031 C75MEX 44197220 IC50 < 1000 nM T79031 CJ8DS1 44198935 IC50 = 42 nM T79031 C0WYG4 44218351 IC50 = 350 nM T79031 CFN2M5 44218508 IC50 = 1800 nM T79031 C8WX5Q 44218512 IC50 = 63 nM T79031 CUFW17 44218800 IC50 = 3200 nM T79031 CV3MJ9 44218957 IC50 = 3400 nM T79031 C7XNT3 44219272 IC50 = 470 nM T79031 C7T1GU 44219759 IC50 = 1100 nM T79031 CZ85SD 44236883 IC50 > 250000 nM T79031 CCJN58 44236884 IC50 > 250000 nM T79031 CZIF43 44236885 Ki = 150000 nM T79031 CC83SD 44236886 IC50 > 250000 nM T79031 C85DAM 44236887 Ki = 64000 nM T79031 C15SQV 44236888 IC50 > 250000 nM T79031 CNB0E9 44236889 IC50 > 250000 nM T79031 C6DR4L 44236890 IC50 > 250000 nM T79031 C6N2KH 44236891 IC50 > 250000 nM T79031 C43UTJ 44247586 Ki = 15 nM T79031 C6HC9D 44258296 IC50 = 5300 nM T79031 CS7XD6 44285533 IC50 = 16 nM T79031 CT62DI 44285546 IC50 = 84 nM T79031 C2V8QE 44285579 IC50 = 55 nM T79031 C1FTJ9 44285580 IC50 = 3.4 nM T79031 CWYC30 44295917 IC50 = 50000 nM T79031 CP23GE 44296131 IC50 = 94000 nM T79031 CFN7R4 44296253 IC50 = 17000 nM T79031 CK9U5X 44296283 IC50 = 11000 nM T79031 C6O5IK 44296284 IC50 = 6000 nM T79031 CG1BS7 44296298 IC50 = 14000 nM T79031 C82TJU 44296317 IC50 = 56000 nM T79031 C2M8IK 44296358 IC50 = 120 nM T79031 C95ZMY 44296370 IC50 = 140000 nM T79031 CP83XL 44296371 IC50 = 130000 nM T79031 CB98RA 44296372 IC50 = 42000 nM T79031 C13DXP 44296399 IC50 > 100000 nM T79031 CWPB94 44296415 IC50 = 48000 nM T79031 CCS9M6 44296416 IC50 = 25000 nM T79031 CP23MY 44296436 IC50 = 4000 nM T79031 CAG4Y2 44296440 IC50 > 200000 nM T79031 C1ZEV5 44296441 IC50 = 4000 nM T79031 CZJ29N 44296442 IC50 = 3000 nM T79031 C74APQ 44296445 IC50 = 10000 nM T79031 CJ9W7L 44296453 IC50 = 4000 nM T79031 C3LDX6 44296454 IC50 = 30000 nM T79031 C53MJG 44296483 IC50 = 47000 nM T79031 C3NVE7 44296484 IC50 = 94000 nM T79031 CZ8AM2 44296485 IC50 > 200000 nM T79031 C5LGI1 44296509 IC50 > 200000 nM T79031 CMP82O 44296586 IC50 = 41000 nM T79031 CHC69E 44296587 IC50 = 28000 nM T79031 C7WVH9 44296588 IC50 = 27000 nM T79031 CKS04O 44296589 IC50 = 28000 nM T79031 CO0V4Y 44296609 IC50 = 47000 nM T79031 C04ICV 44296651 IC50 = 300 nM T79031 C5W2SN 44296652 IC50 = 5000 nM T79031 CC75FT 44296653 IC50 > 100000 nM T79031 C31NFG 44305352 Ki = 68 nM T79031 C0Q3PJ 44305353 Ki = 10 nM T79031 CH6XK9 44305484 Ki = 1129 nM T79031 C8YR3A 44305509 Ki = 0.32 nM T79031 CJ0Y3S 44305543 Ki = 5808 nM T79031 CW7K4A 44305827 Ki = 22423 nM T79031 CDJF28 44305828 Ki = 3134 nM T79031 C26ZWB 44305867 Ki = 8 nM T79031 CU09HP 44305868 Ki = 2.5 nM T79031 C8FG4M 44305869 Ki = 9.4 nM T79031 CX6H1O 44305870 Ki = 5.9 nM T79031 CS0D3M 44305918 Ki = 61.4 nM T79031 CIML79 44305946 Ki = 50.1 nM T79031 C89TJY 44317758 IC50 = 63 nM T79031 C8S3EJ 44317881 IC50 = 75 nM T79031 CA1U4Z 44317882 IC50 = 41 nM T79031 CYS94L 44318039 IC50 = 650 nM T79031 CRK2D7 44318040 IC50 = 419 nM T79031 C5B7LE 44318042 IC50 = 705 nM T79031 C8JTV2 44318044 IC50 = 118 nM T79031 C4PJ7Q 44318059 IC50 = 89000 nM T79031 C1ZU7D 44318060 IC50 = 2530 nM T79031 CGX65H 44318082 IC50 = 4490 nM T79031 C6VRO9 44318083 IC50 = 3180 nM T79031 C4LQ6S 44318084 IC50 = 67 nM T79031 CF4V8H 44318087 IC50 = 190 nM T79031 CSEF87 44318091 IC50 = 60 nM T79031 C6YD4G 44318092 IC50 = 37 nM T79031 CVET20 44318125 IC50 = 230 nM T79031 CANT46 44318126 IC50 = 220 nM T79031 C6TX4I 44318136 IC50 = 176 nM T79031 C1XUQ0 44318137 IC50 = 45 nM T79031 C7U6HZ 44318138 IC50 = 100 nM T79031 CCJ7L9 44318140 IC50 = 4640 nM T79031 CDQ06A 44318141 IC50 = 550 nM T79031 CES4I1 44318142 IC50 = 1740 nM T79031 CL9YX1 44321855 IC50 = 500 nM T79031 C2I4MG 44321943 IC50 > 150000 nM T79031 CXR50K 44321972 IC50 = 1000 nM T79031 CVK6R5 44322068 IC50 > 200000 nM T79031 CCEI08 44322114 IC50 = 5000 nM T79031 CXOB42 44322127 IC50 = 5000 nM T79031 CQF6E7 44322157 IC50 = 500 nM T79031 CEN5G9 44322158 IC50 > 100000 nM T79031 CLX4K3 44322189 IC50 = 300 nM T79031 CHW3K7 44322206 IC50 = 15000 nM T79031 C3KV7J 44322208 IC50 = 20 nM T79031 C6LG8H 44322212 IC50 > 100000 nM T79031 C0QXP6 44329197 Ki = 1.6 nM T79031 CK4I8E 44329209 Ki = 36 nM T79031 CRV13M 44343242 IC50 = 670 nM T79031 CBW34U 44343266 IC50 = 460 nM T79031 CRS8T2 44343292 IC50 = 1300 nM T79031 C2K0DX 44343293 IC50 = 42000 nM T79031 CS9VH2 44343294 IC50 = 9000 nM T79031 C9YXQ7 44343317 IC50 = 34000 nM T79031 CG90MS 44343400 IC50 = 5600 nM T79031 CK3BU4 44343498 IC50 > 100000 nM T79031 C3ZWG2 44343583 IC50 > 100000 nM T79031 CA7IN5 44350821 IC50 > 160000 nM T79031 C9HUE1 44357171 IC50 = 530 nM T79031 C8CAU2 44357172 IC50 > 91000 nM T79031 CX34RF 44357199 IC50 = 1400 nM T79031 COWN52 44357237 IC50 > 91000 nM T79031 CO80YU 44357330 IC50 > 91000 nM T79031 CZ1FB6 44357333 IC50 > 91000 nM T79031 CM2DJ4 44357334 IC50 = 890 nM T79031 C7LT2C 44357361 IC50 = 520 nM T79031 COE56N 44357362 IC50 = 3800 nM T79031 CSM9A6 44357363 IC50 = 830 nM T79031 C0C9RZ 44357454 IC50 = 110 nM T79031 C6SIA3 44357455 IC50 = 140 nM T79031 C9A2YH 44357540 IC50 = 9400 nM T79031 CQ4F5K 44357541 IC50 = 110 nM T79031 C1ELI8 44357569 IC50 = 58 nM T79031 CR4FT3 44361151 EC50 = 10000 nM T79031 CDWH71 44361152 IC50 = 120 nM T79031 CK07AQ 44370533 Ki = 2700 nM T79031 CFB98M 44370558 Ki = 69500 nM T79031 CA2C1S 44370759 Ki = 1900 nM T79031 CMH4K5 44391689 Ki = 26.6 nM T79031 CQ2GR8 44392157 IC50 = 84 nM T79031 CRT7P4 44394717 Ki = 22423 nM T79031 CLO06R 44394718 Ki = 3134 nM T79031 CV8T1W 44394719 Ki = 1129 nM T79031 CZI58M 44394812 Ki = 0.32 nM T79031 CV42IL 44396890 Ki = 22423 nM T79031 CF8N5W 44397017 Ki = 58.8 nM T79031 CGK16Z 44397035 Ki = 3134 nM T79031 CU12IO 44397063 Ki = 1129 nM T79031 C6AG8D 44397069 Ki = 50.1 nM T79031 CL3CD4 44397090 Ki = 61.4 nM T79031 CKAC78 44397092 Ki = 2.5 nM T79031 C2EV9T 44397166 Ki = 9.4 nM T79031 C95WSF 44397171 Ki = 10491 nM T79031 C8E2XZ 44397237 Ki = 5.9 nM T79031 CU0TR3 44397265 Ki = 1.6 nM T79031 CK1M7Y 44397298 Ki = 8 nM T79031 C97GKY 44405960 IC50 = 65 nM T79031 C6MV9A 44410063 IC50 = 1000 nM T79031 C4AKM9 44410069 IC50 = 1600 nM T79031 CC0YZ2 44410070 IC50 = 2600 nM T79031 CJE18M 44410123 IC50 = 3500 nM T79031 CFT4R0 44410174 IC50 = 1700 nM T79031 C2IU1Y 44410240 IC50 = 1700 nM T79031 CP2MV9 44410282 IC50 = 1130 nM T79031 CXJN05 44410285 IC50 = 1900 nM T79031 C80IXJ 44410528 IC50 = 6.4 nM T79031 CS2FA3 44410934 IC50 = 6.4 nM T79031 C95UYM 44413194 IC50 = 17200 nM T79031 C2ZHK3 44413211 IC50 = 20 nM T79031 C2BPF5 44413559 IC50 = 3800 nM T79031 C4PW0V 44413924 IC50 = 20300 nM T79031 CD62TC 44413943 IC50 = 510 nM T79031 CJV8O2 44413944 IC50 = 1120 nM T79031 C1NY7V 44414701 IC50 = 3.3 nM T79031 C5GTM7 44414739 IC50 = 26 nM T79031 CIU9T2 44414827 IC50 = 6.5 nM T79031 CZP7F3 44420106 IC50 = 750 nM T79031 CXC57A 44421346 IC50 = 15 nM T79031 CA71VT 44421347 IC50 = 1180 nM T79031 CBQ57P 44426031 IC50 = 100 nM T79031 C04GKL 44426032 IC50 = 100 nM T79031 CBLF97 44426033 IC50 = 90 nM T79031 CZH59K 44426035 IC50 = 360 nM T79031 CPY4W3 44426036 IC50 = 770 nM T79031 CVG7S6 44426039 IC50 = 1900 nM T79031 CJ2PI1 44426041 IC50 = 250 nM T79031 C4OZ6F 44426043 IC50 = 5 nM T79031 CP80YT 44426045 IC50 = 300 nM T79031 C12NXL 44426048 IC50 = 70 nM T79031 C25NTL 44426051 IC50 = 132 nM T79031 C6G2TH 44426295 IC50 = 350 nM T79031 CJC46Q 44426296 IC50 = 14 nM T79031 C0OP4C 44426297 IC50 = 34 nM T79031 CJQV34 44426298 IC50 = 12 nM T79031 CS1ZO4 44426299 IC50 = 18 nM T79031 CWRV02 44427628 Ki = 30 nM T79031 CV5Q2R 44429035 IC50 = 675 nM T79031 CWA34C 44429036 IC50 = 2020 nM T79031 CJ94BD 44430088 EC50 = 14 nM T79031 C61ERA 44430089 EC50 = 19 nM T79031 CU62AV 44430090 EC50 = 11 nM T79031 CRHO67 44430091 EC50 = 76 nM T79031 C27HKY 44430092 EC50 = 48 nM T79031 C4RQ8C 44430093 EC50 = 59 nM T79031 C2DI8G 44430095 EC50 = 9 nM T79031 CV2IX0 44430096 EC50 = 1 nM T79031 CJDT19 44430097 IC50 = 3 nM T79031 C7Y4QZ 44430104 EC50 = 4 nM T79031 C3ICA4 44430105 EC50 = 24 nM T79031 CYX6D9 44430106 EC50 = 5 nM T79031 CX2YD8 44430109 EC50 = 4 nM T79031 CK71ZC 44433593 IC50 = 2 nM T79031 CA9YC3 44433596 IC50 = 3700 nM T79031 C8Z2UT 44433597 IC50 = 15000 nM T79031 C3AFH5 44433601 IC50 = 400 nM T79031 CS49VX 44433602 IC50 = 13000 nM T79031 CB9Y4K 44433603 IC50 = 22000 nM T79031 C9ZVY2 44433604 IC50 = 6000 nM T79031 CA9O8Z 44433605 IC50 = 1800 nM T79031 C6RE0Q 44433606 IC50 = 7000 nM T79031 C2VWG1 44433607 IC50 = 15000 nM T79031 C1GSB2 44434133 IC50 = 30000 nM T79031 CD57ZN 44434773 IC50 = 1540 nM T79031 C4VF0U 44434774 IC50 = 1550 nM T79031 CE1KR3 44434775 IC50 = 140 nM T79031 C2QAP8 44434776 IC50 = 280 nM T79031 CU4B2Y 44441701 IC50 = 17 nM T79031 C6QMY7 44441703 IC50 = 2 nM T79031 C0GEN7 44441704 IC50 = 49 nM T79031 CW6BL8 44441705 IC50 = 12 nM T79031 C4QZ5V 44441708 IC50 = 1 nM T79031 CKS0R9 44441710 IC50 = 56 nM T79031 C8ZB2V 44441713 IC50 = 196 nM T79031 CC9J8U 44441716 IC50 = 10 nM T79031 C01SGJ 44441718 IC50 = 290 nM T79031 CG3C1F 44441721 IC50 = 85 nM T79031 CAU32P 44441725 IC50 = 175 nM T79031 C5FEJ8 44441727 IC50 = 53 nM T79031 CR0NY5 44441729 IC50 = 1100 nM T79031 CC35XR 44441732 IC50 = 16 nM T79031 CTC94G 44441736 IC50 = 38 nM T79031 CR74JU 44441738 IC50 = 4 nM T79031 CLJ1R7 44441740 IC50 = 270 nM T79031 C8IB2Z 44441742 IC50 = 780 nM T79031 C2JE8M 44441743 IC50 = 27 nM T79031 C29IKL 44441744 IC50 = 130 nM T79031 CRH2E8 44441745 IC50 = 46 nM T79031 C24HDJ 44441746 IC50 = 78 nM T79031 C3PR7Y 44441747 IC50 = 22 nM T79031 C6SU2Z 44441748 IC50 = 46 nM T79031 CYBA49 44445141 IC50 = 4100 nM T79031 C6G8VL 44445142 IC50 > 20000 nM T79031 C31TEH 44445143 IC50 = 5214 nM T79031 C97WEK 44445144 IC50 > 20000 nM T79031 C47PWX 44445145 IC50 = 3670 nM T79031 C7I0VE 44445146 IC50 > 20000 nM T79031 CDWQ62 44445147 IC50 > 20000 nM T79031 CX50FP 44445148 IC50 = 5614 nM T79031 CX6IA7 44445149 IC50 = 314 nM T79031 C4FRC0 44445150 IC50 = 6461 nM T79031 CC3Z0V 44445151 IC50 = 3785 nM T79031 C1XRF3 44445152 IC50 = 5015 nM T79031 CXH12K 44445153 IC50 = 1090 nM T79031 CTH2D6 44445154 IC50 = 7950 nM T79031 CFQ21V 44445155 IC50 = 484 nM T79031 C68VFD 44446196 IC50 = 5400 nM T79031 C4S1CA 44446197 IC50 = 1120 nM T79031 C7K1RZ 44446198 IC50 = 650 nM T79031 C5CS2Z 44446199 IC50 = 5890 nM T79031 CZO7A4 44446200 IC50 = 33 nM T79031 CJVG08 44446201 IC50 = 550 nM T79031 CF7RP8 44446202 IC50 = 790 nM T79031 CU54SK 44446203 IC50 = 17 nM T79031 CJ3BD7 44446204 IC50 = 1700 nM T79031 CJW16S 44446205 IC50 = 600 nM T79031 CSPE84 44446206 IC50 = 160 nM T79031 CS42CJ 44446207 IC50 = 34670 nM T79031 C7VX1Q 44446209 IC50 = 83 nM T79031 CG4N8T 44446210 IC50 = 100 nM T79031 C1HZ9O 44446211 IC50 = 330 nM T79031 CN2AB7 44446212 IC50 = 230 nM T79031 COQR59 44446520 Ki = 564 nM T79031 CZ6HW7 44446521 Ki = 230 nM T79031 C9QS2X 44446522 Ki = 27 nM T79031 CP02CD 44446523 Ki = 617 nM T79031 C0L3BP 44446524 Ki = 916 nM T79031 C1R6BA 44446525 Ki = 425 nM T79031 CNA92X 44446526 Ki = 552 nM T79031 CP7S1R 44446527 Ki = 894 nM T79031 CY5D4A 44446528 Ki = 15000 nM T79031 CX1ZM5 44446545 Ki = 0.12 nM T79031 CI6K3D 44447213 IC50 = 3000 nM T79031 CQI94E 44447217 IC50 = 4600 nM T79031 C5ZP8F 44447252 IC50 = 3500 nM T79031 CH6G1V 44447299 IC50 = 5750 nM T79031 CJ10US 44447357 IC50 = 600 nM T79031 CKFT76 44447358 IC50 = 800 nM T79031 C9FN0P 44447372 IC50 = 2000 nM T79031 CG5C1R 44447389 IC50 = 2000 nM T79031 CFC0T1 44447406 IC50 = 500 nM T79031 CW21CI 44447407 IC50 = 600 nM T79031 CDZF34 44447421 IC50 = 600 nM T79031 CMX0B6 44447422 IC50 = 900 nM T79031 CT3S5H 44447454 IC50 = 700 nM T79031 CW0LK4 44449760 Ki = 1256 nM T79031 C5LJY9 44449874 Ki = 662 nM T79031 CHU63Z 44449992 Ki = 6800 nM T79031 C34HBT 44450018 Ki = 39989 nM T79031 C7GQY6 44450048 Ki = 3005 nM T79031 CL1SO0 44450074 Ki = 2194 nM T79031 C0GOH4 44450139 Ki = 9 nM T79031 C0EPX3 44450198 Ki = 18 nM T79031 C2PJ1L 44450200 Ki = 1881 nM T79031 CXS7Y3 44454508 IC50 = 59 nM T79031 C2QI1J 44454509 IC50 = 745 nM T79031 CML29V 44454541 IC50 = 5270 nM T79031 CBS73X 44454542 IC50 = 62000 nM T79031 CJ0NI6 44454543 IC50 = 1900 nM T79031 CW2LM3 44454574 IC50 > 500000 nM T79031 C6XF5J 44454575 IC50 > 500000 nM T79031 CQ5JM2 44454576 IC50 > 500000 nM T79031 C6NC4X 44454662 IC50 = 29.9 nM T79031 C0XMF7 44454839 IC50 = 72 nM T79031 CTY3G5 44454842 IC50 = 860 nM T79031 CIFD60 44454874 IC50 = 39 nM T79031 CP08GW 44454875 IC50 = 180 nM T79031 CU9GD7 44454913 IC50 = 1450 nM T79031 C6XY2B 44454914 IC50 = 605 nM T79031 C7OGW4 44454944 IC50 = 120 nM T79031 C10PVS 44454945 IC50 = 32 nM T79031 CO8M3N 44455060 IC50 = 780 nM T79031 CT9N4O 44455061 IC50 = 89 nM T79031 CAMP21 44455062 IC50 = 65 nM T79031 CC7JN8 44455094 IC50 = 770 nM T79031 CR2VQ6 44455207 IC50 = 26 nM T79031 CS03JA 44455208 IC50 = 12 nM T79031 C1KOX9 44455269 IC50 = 120 nM T79031 CWS72U 44455302 IC50 = 630 nM T79031 CO3TS7 44455303 IC50 = 2000 nM T79031 CXON46 44455334 IC50 = 191 nM T79031 C5S1WG 44455335 IC50 = 4200 nM T79031 C8QVZ3 44455369 IC50 = 1350 nM T79031 C14FHC 44455370 IC50 = 330 nM T79031 CG12UX 44455371 IC50 = 440 nM T79031 C7NM8F 44455390 IC50 = 70 nM T79031 CX7F4D 44455419 IC50 = 240 nM T79031 C9SB5E 44455462 IC50 = 293 nM T79031 CI7GZ9 44455467 IC50 = 365 nM T79031 C1A9TW 44455472 IC50 = 321 nM T79031 CCQ05S 44455474 IC50 = 203 nM T79031 C24BWX 44455486 IC50 = 570 nM T79031 CZSO57 44455487 IC50 = 295 nM T79031 C6YB9L 44455500 IC50 = 137 nM T79031 CWTH48 44455501 IC50 = 124 nM T79031 C5A7CY 44455514 IC50 = 110 nM T79031 CEKI49 44455515 IC50 = 57 nM T79031 CY68NV 44455516 IC50 = 78 nM T79031 C7WCZ8 44455529 IC50 = 278 nM T79031 C6MX9L 44455530 IC50 = 172 nM T79031 CU07LG 44455531 IC50 = 130 nM T79031 CLT1R8 44455543 IC50 = 142 nM T79031 CL9N0S 44455544 IC50 = 1200 nM T79031 C1EWG9 44455554 IC50 = 125 nM T79031 CJ3V2W 44455567 IC50 = 303 nM T79031 CI34FJ 44455570 IC50 = 225 nM T79031 CS2HG8 44455573 IC50 = 219 nM T79031 CR9V2G 44455581 IC50 = 78 nM T79031 CGW49Q 44455601 IC50 = 365 nM T79031 CD7GY0 44455602 IC50 = 312 nM T79031 CYQM64 44455636 IC50 = 46000 nM T79031 CN3JK0 44455638 IC50 = 338 nM T79031 C1VD5W 44455639 IC50 = 350 nM T79031 CAQ03Z 44455666 IC50 = 2800 nM T79031 C8GC4O 44455667 IC50 = 18800 nM T79031 CQFW59 44455691 IC50 = 850 nM T79031 C2A6DO 44455692 IC50 = 290 nM T79031 CS16QI 44455695 IC50 = 270 nM T79031 C6X9DY 44455721 IC50 = 2950 nM T79031 C5HQN3 44455724 IC50 = 2000 nM T79031 C1FM6T 44455733 IC50 = 7200 nM T79031 CGK5A1 44455750 IC50 = 155 nM T79031 CT8QL3 44455753 IC50 = 100 nM T79031 CU0NA7 44455754 IC50 = 71 nM T79031 C3X7BU 44455772 IC50 = 45 nM T79031 CJ4I3V 44455775 IC50 = 370 nM T79031 COL9T5 44455798 IC50 = 3000 nM T79031 CH8IB5 44455802 IC50 = 900 nM T79031 CZY7I2 44455803 IC50 = 7000 nM T79031 CF9ZC6 44455830 IC50 = 651 nM T79031 CX2BH5 44455859 IC50 = 558 nM T79031 C34BAL 44455860 IC50 = 203 nM T79031 CD7U9X 44455861 IC50 = 752 nM T79031 C3FJ5Z 44455881 IC50 = 269 nM T79031 C14YKA 44455882 IC50 = 241 nM T79031 CZUW95 44455900 IC50 = 149 nM T79031 CC1M7L 44455901 IC50 = 116 nM T79031 CIQ06V 44456429 IC50 = 121 nM T79031 CV0A2R 44456430 IC50 = 114 nM T79031 CKN04W 44456431 IC50 = 151 nM T79031 CYVS69 44456474 IC50 = 133 nM T79031 CINB34 44456475 IC50 = 150 nM T79031 CD0V2B 44460227 IC50 = 70 nM T79031 CV6K1D 44460349 IC50 = 28 nM T79031 C8HSO1 44460350 IC50 = 127 nM T79031 C8GYW2 44462104 IC50 = 1130 nM T79031 CL61RT 44462105 IC50 = 350 nM T79031 C46PUO 44462123 IC50 = 350 nM T79031 CG96TF 44462737 IC50 = 1300 nM T79031 C7UDS1 44467360 Ki = 5 nM T79031 C8C1VG 44467504 Ki = 8 nM T79031 C0CNQ3 44467506 Ki = 20 nM T79031 CL5XQ6 44467507 Ki = 36 nM T79031 C41RNH 44467574 Ki = 8.5 nM T79031 C8TIU2 44467575 Ki = 6 nM T79031 CM41YP 44467576 Ki = 7 nM T79031 CLU19G 44467711 Ki = 30 nM T79031 CVC68I 44467853 Ki = 53 nM T79031 CAGM05 44478390 IC50 = 190 nM T79031 C9P3XR 44478656 IC50 = 80 nM T79031 CA4W3P 44478657 EC50 = 3000 nM T79031 CX24EA 44478658 EC50 = 1600 nM T79031 CJ7AL5 44478659 IC50 = 160 nM T79031 CC3VB8 44478660 IC50 = 740 nM T79031 CY4MJ6 44478726 Ki = 10 nM T79031 CD5X8P 44478997 Ki = 11 nM T79031 C6Q8JT 44479264 Ki = 15 nM T79031 CP64VM 44479524 Ki = 48 nM T79031 CW8Z4Q 44480205 Ki = 211 nM T79031 CA2T1B 44480209 Ki = 295 nM T79031 CG5D2O 44514457 IC50 = 710 nM T79031 C9S7OU 44514742 IC50 = 100 nM T79031 C4F0AI 44514744 IC50 = 290 nM T79031 CTKE78 44515351 IC50 = 1500 nM T79031 CI2X9B 44517765 IC50 = 230 nM T79031 C8QT4P 44517766 IC50 = 250 nM T79031 C1R7BX 44552610 IC50 = 250000 nM T79031 C0W4MU 44563122 IC50 = 36800 nM T79031 CCO70V 44570172 IC50 = 1581 nM T79031 CMNO27 44570173 IC50 = 2506 nM T79031 C26UXD 44570174 IC50 = 889 nM T79031 C9JI2N 44570207 IC50 = 2233 nM T79031 C0CFU7 44570208 IC50 = 811 nM T79031 CCN7P9 44570209 IC50 = 1119 nM T79031 CL8SM0 44570210 IC50 = 1256 nM T79031 CVW7F2 44570211 IC50 = 1774 nM T79031 C34VYL 44570212 IC50 = 158 nM T79031 C78FBX 44570213 IC50 = 524 nM T79031 CSE6U7 44570261 IC50 = 740 nM T79031 COI30F 44570262 IC50 = 262 nM T79031 CJ2MR9 44570263 IC50 = 998 nM T79031 CTB4F0 44570302 IC50 = 112 nM T79031 C1Q0DR 44570303 IC50 = 89 nM T79031 CVP9O4 44570540 IC50 = 47090 nM T79031 C48ZIJ 44582543 Ki = 0.8 nM T79031 C6PL5S 44586336 IC50 = 2 nM T79031 CCL36O 44586337 IC50 = 57 nM T79031 CVW0L1 44586338 IC50 = 9 nM T79031 CZ9I7T 44586406 IC50 = 905 nM T79031 CLXV20 44586407 IC50 = 180 nM T79031 C9RX5T 44586408 IC50 = 140 nM T79031 CA4J5W 44586409 IC50 = 3 nM T79031 CK6T1E 44586453 IC50 = 88 nM T79031 CR82MH 44586454 IC50 = 16 nM T79031 CHF74X 44586455 IC50 = 1400 nM T79031 C8IF6Q 44586456 IC50 = 13 nM T79031 CO4P6S 44586494 IC50 = 9 nM T79031 CMZ04I 44586495 IC50 = 11 nM T79031 CI2P0W 44586496 IC50 = 790 nM T79031 CH2X1J 44586497 IC50 = 7500 nM T79031 CU5ZE8 44586498 IC50 = 235 nM T79031 C8TUY6 44586534 IC50 = 175 nM T79031 CPC5H1 44586535 IC50 = 44 nM T79031 C53LNK 44586536 IC50 = 13 nM T79031 CDAM25 44586537 IC50 = 915 nM T79031 C0Y3SP 44586538 IC50 = 5 nM T79031 C3QXF2 44586539 IC50 = 20 nM T79031 CIR8Y3 44586540 IC50 = 27 nM T79031 CN65TC 44586541 IC50 = 345 nM T79031 CTA78Q 44588631 IC50 > 10000 nM T79031 C5L4NQ 44588632 IC50 > 10000 nM T79031 C2E4RJ 44588633 IC50 = 200 nM T79031 CQ18CM 44588634 IC50 = 14 nM T79031 C4WXC8 44588635 IC50 = 120 nM T79031 C3WC1U 44588636 IC50 = 24 nM T79031 CG42IK 44588637 IC50 = 1200 nM T79031 CQAT24 44588638 IC50 = 220 nM T79031 CF0N6C 44588639 IC50 = 40 nM T79031 CA6I3V 44588640 IC50 = 2230 nM T79031 C8DB1H 44588641 IC50 = 1890 nM T79031 CA5SD6 44588642 IC50 = 1600 nM T79031 C3JY7V 44588643 IC50 > 10000 nM T79031 C9LZ3U 44588644 IC50 = 4000 nM T79031 CKEZ47 44588645 IC50 = 2300 nM T79031 CB1Q4T 44588646 IC50 = 210 nM T79031 CFY78K 44588647 IC50 = 260 nM T79031 CLF0E5 44588648 IC50 > 10000 nM T79031 C5W7KN 44588649 IC50 > 10000 nM T79031 CP3V1I 44590652 IC50 < 1000 nM T79031 CF32HV 44590653 IC50 < 1000 nM T79031 C8FW1J 44590654 IC50 < 1000 nM T79031 C46PHY 44590655 IC50 < 1000 nM T79031 CPA8Y6 44590656 IC50 < 1000 nM T79031 CTZ1I6 44590657 IC50 < 1000 nM T79031 C7G9BS 44590658 IC50 < 1000 nM T79031 CQ3W8L 44590659 IC50 < 1000 nM T79031 C0G7RS 44590660 IC50 < 1000 nM T79031 C1YDI4 44590661 IC50 = 54.6 nM T79031 C4WVO3 44590662 IC50 = 771 nM T79031 CA7B1X 44590663 IC50 < 1000 nM T79031 C8F1HZ 44591546 IC50 = 22 nM T79031 CG32VI 44591547 IC50 = 15 nM T79031 CRA23E 44591548 IC50 = 24 nM T79031 CEPV57 44591549 IC50 = 13 nM T79031 CB15AK 44591550 IC50 = 9 nM T79031 C9Q7TN 44591551 IC50 = 10 nM T79031 CNIX24 44592569 IC50 = 35000 nM T79031 CL1PQ6 44604353 IC50 > 10000 nM T79031 C34RFE 44604423 IC50 = 310 nM T79031 C3E5AZ 44624107 IC50 = 78 nM T79031 CUIY75 44624171 IC50 = 40 nM T79031 CT46YX 44624237 IC50 = 100 nM T79031 C8A2VT 44624238 IC50 = 118 nM T79031 CT65UM 44624240 IC50 = 6 nM T79031 C6N3JL 44624304 IC50 = 61 nM T79031 C7AB0L 44625098 IC50 = 49 nM T79031 C5WU0H 44625099 IC50 = 2 nM T79031 CL4BZ5 44625321 IC50 = 346 nM T79031 C9ZGM1 44625323 IC50 = 4 nM T79031 CIO27W 44625397 IC50 = 126 nM T79031 CGX41M 44631838 IC50 = 0.32 nM T79031 CHL19P 44631842 IC50 = 17 nM T79031 CQ9G6O 44631933 IC50 = 10 nM T79031 CF9TI0 45105269 IC50 = 1150 nM T79031 C87CZK 45105273 Ki = 3 nM T79031 C3M7ZG 45105274 Ki = 0.8 nM T79031 C9CK4G 45112084 IC50 > 10000 nM T79031 C5DQK2 45112086 IC50 = 1860 nM T79031 C4M9OX 45112223 IC50 = 6500 nM T79031 CJ85ZC 45112224 IC50 = 1500 nM T79031 C5G7ID 45112225 IC50 = 2030 nM T79031 CKF82L 45112226 IC50 > 10000 nM T79031 C36HCE 45112334 IC50 > 10000 nM T79031 CF1P7X 45112335 IC50 = 240 nM T79031 C1JNV3 45112336 IC50 = 140 nM T79031 C6QPX4 45112337 IC50 = 1500 nM T79031 CEO74L 45112444 IC50 > 10000 nM T79031 C0Z4CY 45112445 IC50 > 10000 nM T79031 C9EKY3 45114034 IC50 = 1500 nM T79031 CI8P2O 45114035 IC50 > 10000 nM T79031 CJ0Y1O 45254127 IC50 = 0.7 nM T79031 C8FQ9P 45254130 IC50 = 0.6 nM T79031 CQB45G 45254505 IC50 = 2.5 nM T79031 C1R3PL 45254506 IC50 = 2.5 nM T79031 C2JD1Y 45254508 IC50 = 7.1 nM T79031 C2YE7A 45254510 IC50 = 0.7 nM T79031 C87CFA 45254702 IC50 = 0.4 nM T79031 C2M9RC 45254900 IC50 = 4 nM T79031 CUL8G3 45255106 IC50 = 3 nM T79031 CK76PW 45255111 IC50 = 5.4 nM T79031 CF92SD 45255915 IC50 = 52 nM T79031 CA5YG0 45256104 IC50 = 107 nM T79031 C0H9YA 45256107 IC50 = 1430 nM T79031 CRB2J3 45256108 IC50 = 740 nM T79031 C43HDC 45256109 IC50 = 25 nM T79031 C2Q3MJ 45256294 IC50 = 8 nM T79031 C5RQ2B 45256296 IC50 = 3.1 nM T79031 C0Q2WV 45256478 IC50 = 8 nM T79031 C8H4SQ 45256479 IC50 = 4 nM T79031 CGC2A0 45256481 IC50 = 15 nM T79031 CV32EW 45256653 IC50 = 4 nM T79031 C5LYK1 45256654 IC50 = 19 nM T79031 CE9IU1 45256823 IC50 = 2 nM T79031 CI70YH 45256826 IC50 = 4.5 nM T79031 CT41IW 45256827 IC50 = 30 nM T79031 C61DTC 45259043 IC50 = 53 nM T79031 C8BYZ2 45259044 IC50 = 3700 nM T79031 C52YGJ 45267231 IC50 = 198 nM T79031 CR28KS 45267235 IC50 = 52 nM T79031 C0JR5F 45267240 IC50 = 12 nM T79031 CIY5X1 45267880 IC50 = 28 nM T79031 C97DIE 45268098 IC50 = 122 nM T79031 CXBU68 45268099 IC50 = 137 nM T79031 CZ7R3C 45268100 IC50 = 12 nM T79031 C0LPK9 45268101 IC50 = 10 nM T79031 C4SDU6 45268102 IC50 = 30 nM T79031 CTS4W8 45268589 IC50 > 10000 nM T79031 C1LYC5 45268590 IC50 = 2500 nM T79031 CD2MC1 45268670 IC50 = 86 nM T79031 CFA5L4 45268963 IC50 = 20 nM T79031 CS1ND7 45268964 IC50 = 166 nM T79031 C05MYF 45268967 IC50 = 25 nM T79031 C2LON9 45268972 IC50 = 148 nM T79031 CV0J8R 45269443 IC50 = 4000 nM T79031 C8WGE2 45269491 IC50 = 12 nM T79031 C16WVK 45269615 IC50 = 490 nM T79031 C94IYG 45269822 IC50 = 51 nM T79031 CCPJ13 45269826 IC50 = 43 nM T79031 CP63SL 45269828 IC50 = 151 nM T79031 C7IGC0 45270281 IC50 > 10000 nM T79031 CD0GT7 45270282 IC50 = 450 nM T79031 CLPZ81 45270645 IC50 = 10 nM T79031 C0RJ1K 45270646 IC50 = 168 nM T79031 CP6R4L 45270650 IC50 = 74 nM T79031 CS8F0K 45270651 IC50 = 90 nM T79031 C9CXR6 45270652 IC50 = 428 nM T79031 C6R9HW 45270653 IC50 = 31 nM T79031 CH9W5L 45270656 IC50 = 173 nM T79031 CL1EZ9 45270657 IC50 = 184 nM T79031 C40TXF 45271106 IC50 = 5900 nM T79031 CPN7C0 45271107 IC50 > 10000 nM T79031 C08VIR 45271108 IC50 = 4600 nM T79031 C78TLW 45271466 IC50 = 55 nM T79031 CJC68W 45271467 IC50 = 123 nM T79031 CDVI91 45271468 IC50 = 92 nM T79031 C0EV5Y 45271469 IC50 = 32 nM T79031 C67OZF 45271474 IC50 = 59 nM T79031 CPX16M 45271476 IC50 = 94 nM T79031 C2OHU1 45272371 IC50 = 80 nM T79031 C5I3UC 45272372 IC50 = 67 nM T79031 C8XBJ3 45272373 IC50 = 16 nM T79031 C8ZDL9 45272374 IC50 > 2000 nM T79031 CYQ0K6 45272375 IC50 = 37 nM T79031 C5QWR8 45272378 IC50 = 111 nM T79031 CVW8G1 45272379 IC50 = 124 nM T79031 CMR73U 45272383 IC50 = 52 nM T79031 CY0FT4 45272384 IC50 = 27 nM T79031 CK8H7U 45272385 IC50 = 10 nM T79031 C4L5CK 45272386 IC50 = 54 nM T79031 CRCO14 45272821 IC50 > 10000 nM T79031 CBM78N 45273242 IC50 = 10 nM T79031 C54QPK 45273243 IC50 = 20 nM T79031 C6M3ZT 45273244 IC50 = 86 nM T79031 C5NTQ6 45273245 IC50 = 24 nM T79031 C7L5IK 45273251 IC50 = 75 nM T79031 C8MT1Z 45273255 IC50 = 9 nM T79031 CIUZ85 45273256 IC50 = 242 nM T79031 C2KQ9U 45273257 IC50 = 13 nM T79031 CDCY81 45273772 IC50 = 5600 nM T79031 CVHF18 45273773 IC50 > 10000 nM T79031 C6JFK8 45277565 IC50 = 4500 nM T79031 CVPF48 45277566 IC50 = 10000 nM T79031 C6S2BO 45277567 IC50 = 1260 nM T79031 CJVC29 45277727 IC50 > 10000 nM T79031 C5AWL1 45483144 Ki = 244 nM T79031 C5EF4Y 45483153 Ki = 10 nM T79031 CJ7Q8L 45483165 Ki = 348 nM T79031 C9IV4D 45483169 Ki = 293 nM T79031 CC59XA 45483174 Ki = 309 nM T79031 CL7Q8K 45483917 IC50 = 480 nM T79031 CSY12G 45483918 IC50 = 1800 nM T79031 CJ3WD1 45484135 IC50 = 50000 nM T79031 CYLN37 45484139 IC50 = 3000 nM T79031 CX2D0E 45484151 IC50 = 7000 nM T79031 CL4V7R 45484174 IC50 = 78000 nM T79031 C4JD9S 45484175 IC50 = 5000 nM T79031 CJDC46 45484184 IC50 = 2100 nM T79031 C9MI1Y 45484250 IC50 = 27 nM T79031 C1C6VB 45486934 IC50 > 10000 nM T79031 CF1RV5 45486939 IC50 > 10000 nM T79031 CTX69D 45486942 IC50 = 4700 nM T79031 CD0S3I 45486943 IC50 = 47 nM T79031 CEWV96 45486944 IC50 = 210 nM T79031 C79FXL 45486945 IC50 = 240 nM T79031 CUS3W8 45486946 IC50 = 500 nM T79031 C04CSV 45486950 IC50 = 8.8 nM T79031 C3E5LA 45486952 IC50 = 120 nM T79031 CIM9P8 45486956 IC50 = 380 nM T79031 CRO40Q 45486957 IC50 = 19 nM T79031 CZU54V 45486959 IC50 = 19 nM T79031 C2O9HI 45486960 IC50 = 24 nM T79031 CZDO08 45486961 IC50 = 49 nM T79031 CO24SK 45486962 IC50 = 24 nM T79031 CA2B9J 45486963 IC50 = 350 nM T79031 C5YI3E 45486972 IC50 = 33 nM T79031 CG16NB 45486973 IC50 = 100 nM T79031 CB70SF 45486975 IC50 = 140 nM T79031 CO4NR2 45486979 IC50 = 59 nM T79031 CPYS43 45486980 IC50 = 400 nM T79031 C98DLY 45486981 IC50 = 860 nM T79031 C8E2PU 45486982 IC50 = 380 nM T79031 CROV56 45486983 IC50 = 240 nM T79031 C8JQ7T 45486984 IC50 = 73 nM T79031 C36ZXE 45486988 IC50 = 1300 nM T79031 C1HK5L 45486991 IC50 = 270 nM T79031 CD9IL6 45486996 IC50 = 210 nM T79031 CS5D9N 45486998 IC50 = 220 nM T79031 CS60MQ 45486999 IC50 = 2400 nM T79031 CKO57E 45487000 IC50 = 330 nM T79031 CB3D5J 45487001 IC50 = 85 nM T79031 CF9IZ0 45487004 IC50 = 38 nM T79031 CR90BO 45487005 IC50 = 400 nM T79031 C4NTM7 45488098 EC50 = 70 nM T79031 CT95YJ 45488099 EC50 = 1200 nM T79031 C6W8LK 45488101 IC50 = 469.89 nM T79031 CHMZ65 45488102 EC50 = 230 nM T79031 C4GVA9 45488103 EC50 = 8130 nM T79031 CT51JC 45488104 EC50 = 130 nM T79031 C1Q9DK 45488105 IC50 = 10 nM T79031 CJ13RL 45488106 IC50 = 1390 nM T79031 CH7SG2 45488107 IC50 = 320 nM T79031 CL0H9O 45488108 EC50 = 1900 nM T79031 C9KP7N 45488109 IC50 = 3467.37 nM T79031 CJ75VZ 45488110 IC50 = 1360 nM T79031 C4QV8Z 45488111 IC50 = 59.98 nM T79031 C4ZD5W 45488112 IC50 = 520 nM T79031 CXG2R1 45488113 Ki = 300 nM T79031 C9NG1H 45488114 IC50 = 3097.42 nM T79031 C8FTJ3 45488115 EC50 = 2130 nM T79031 CB10OE 45488116 IC50 = 900 nM T79031 CE1ZX5 45488119 IC50 = 20 nM T79031 CKBT31 45488120 EC50 = 270 nM T79031 CH0W9R 45488121 EC50 = 60 nM T79031 CV84ZK 45489778 IC50 = 460000 nM T79031 COT0P1 46178810 EC50 = 36 nM T79031 CVW76R 46190732 IC50 = 9 nM T79031 CZ0JD1 46191766 IC50 = 70 nM T79031 C5CV9T 46200991 IC50 = 16200 nM T79031 C7VR2G 46202081 IC50 = 86.4 nM T79031 C56SZE 46202415 IC50 = 17 nM T79031 C38LWQ 46202743 IC50 = 2.92 nM T79031 C4A5NH 46203391 IC50 = 3.4 nM T79031 CR0WQ3 46204457 IC50 = 6930 nM T79031 CT3PN7 46204458 IC50 = 15730 nM T79031 C7HTE3 46204763 IC50 = 4670 nM T79031 C6SV7F 46204764 IC50 = 8070 nM T79031 C6DPI0 46205407 IC50 = 3790 nM T79031 C0OWZ3 46205408 IC50 = 2640 nM T79031 CK0Q7W 46205409 IC50 = 3810 nM T79031 C7KRN0 46205733 IC50 = 4240 nM T79031 CQPA53 46205737 IC50 = 2310 nM T79031 C9MPG6 46205967 IC50 = 11.4 nM T79031 CNVX45 46205968 IC50 = 8.25 nM T79031 CR9A5G 46206291 IC50 = 198 nM T79031 C9B1CG 46206292 IC50 = 125 nM T79031 CSX8P1 46206294 IC50 = 137 nM T79031 CD0R7T 46206296 IC50 = 135 nM T79031 CR1X0F 46206642 IC50 = 43.1 nM T79031 C8JYQ3 46206643 IC50 = 10.7 nM T79031 C0R1YT 46206645 IC50 = 29.9 nM T79031 CH8Y7D 46206977 IC50 = 21.5 nM T79031 C51XNJ 46209414 Ki = 98.8 nM T79031 C3VYC6 46217866 IC50 = 800 nM T79031 CH2EI5 46218828 Ki = 0.017 nM T79031 C0V2KN 46218829 Ki > 1000 nM T79031 CM9ON2 46225154 IC50 = 55 nM T79031 CY9O4P 46225190 IC50 = 1080 nM T79031 C1WU7T 46225198 IC50 = 27 nM T79031 CJDR54 46225199 IC50 = 60 nM T79031 C3L5CE 46225200 IC50 = 19 nM T79031 C5KWY2 46225201 IC50 = 1 nM T79031 CJCU20 46225202 IC50 = 668 nM T79031 C0EGN7 46225203 IC50 = 83 nM T79031 CV0PC7 46225204 IC50 = 177 nM T79031 CML6Q8 46225205 IC50 > 10000 nM T79031 CQMD65 46225238 IC50 = 2850 nM T79031 CUP1F4 46225247 IC50 = 1 nM T79031 C1B8SI 46225248 IC50 = 2 nM T79031 CVD16W 46225249 IC50 = 50 nM T79031 CXN95V 46225250 IC50 = 67 nM T79031 C37PUF 46225251 IC50 = 50 nM T79031 CZS8H2 46225290 IC50 = 380 nM T79031 C5XT0R 46229681 IC50 = 185600 nM T79031 C3GD0Y 46229698 IC50 = 203300 nM T79031 CW94EK 46229699 IC50 = 203300 nM T79031 C4O6GY 46231497 IC50 = 69.98 nM T79031 C4NCL1 46231498 IC50 = 150 nM T79031 C51DSC 46231499 IC50 = 300 nM T79031 C1K6QJ 46231500 IC50 = 29.99 nM T79031 CK3O2Q 46231555 IC50 = 10 nM T79031 CY23FV 46231556 IC50 = 10 nM T79031 CIA4F3 46233415 Ki = 60 nM T79031 CJZT40 46233416 Ki = 80 nM T79031 CKE7B8 46233417 Ki = 75 nM T79031 C1EH4N 46233418 Ki < 1 nM T79031 CD6EK4 46233419 Ki = 9 nM T79031 C8HX0R 46233420 Ki = 1800 nM T79031 CF5IV9 46233421 Ki = 400 nM T79031 CPKS32 46233422 Ki = 1400 nM T79031 CD8IS3 46233423 Ki = 200 nM T79031 CETW51 46233424 Ki = 100 nM T79031 CJ96GE 46233425 Ki > 10000 nM T79031 C8IFJ3 46233426 Ki = 220 nM T79031 CU3EI0 46233611 Ki = 20 nM T79031 CO6HY7 46233612 Ki = 1.3 nM T79031 C0B6LM 46233613 Ki = 130 nM T79031 C4IP1B 46233614 Ki = 210 nM T79031 CHA57O 46233615 Ki = 70 nM T79031 CG30XW 46233616 Ki = 140 nM T79031 CU6TZ0 46238535 IC50 = 26000 nM T79031 CZK5E9 46238536 IC50 = 7000 nM T79031 C6UF9A 46239657 Ki = 104 nM T79031 C5ILT9 46239761 Ki = 37.5 nM T79031 C6NE9Y 46369107 IC50 = 100000 nM T79031 CY4SD8 46371748 IC50 = 100000 nM T79031 CI0AP7 46702891 IC50 = 26900 nM T79031 C71PDX 46703353 IC50 = 16100 nM T79031 CODI24 46703649 IC50 = 29300 nM T79031 CN68GQ 46703650 IC50 = 26400 nM T79031 CNO20W 46703651 IC50 = 33100 nM T79031 C2QOL0 46703794 IC50 = 27100 nM T79031 C61FYH 46703795 IC50 = 26600 nM T79031 C6E1IM 46703796 IC50 = 23200 nM T79031 C01IOM 46703955 IC50 = 39100 nM T79031 C81XKI 46703956 IC50 = 28400 nM T79031 CP15OJ 46703957 IC50 = 28200 nM T79031 CL1VG6 46704110 IC50 = 16100 nM T79031 C7ZB2N 46704111 IC50 = 29300 nM T79031 CEK5U7 46704268 IC50 = 26100 nM T79031 CRV1L2 46704273 IC50 = 31900 nM T79031 CVQ9M8 46704412 IC50 = 24600 nM T79031 CQ08BY 46704413 IC50 = 30400 nM T79031 C6KN1D 46830239 IC50 = 20 nM T79031 CNP2S7 46844428 IC50 = 2.5 nM T79031 C7D4SK 46844429 IC50 = 150 nM T79031 CPTV06 46845694 IC50 = 163 nM T79031 CY8S4A 46848865 IC50 = 135000 nM T79031 C8RTV2 46849021 IC50 = 155000 nM T79031 C9U4IE 46849022 IC50 = 82000 nM T79031 CCQA47 46849023 IC50 = 163000 nM T79031 CW9U7P 46849024 IC50 = 90000 nM T79031 CG94IE 46849025 IC50 = 93000 nM T79031 C35KQB 46849026 IC50 = 98000 nM T79031 CJW83F 46849027 IC50 = 104000 nM T79031 CXN3C5 46861631 Ki = 1 nM T79031 CNSO83 46861889 Ki = 1 nM T79031 CA3RK8 46881101 IC50 = 3600 nM T79031 C0LQ8O 46881431 IC50 = 10800 nM T79031 CZ03ED 46881490 IC50 = 22200 nM T79031 C58JMD 46881491 IC50 = 24900 nM T79031 CK5U6I 46881492 IC50 = 580 nM T79031 CR8CP9 46881519 IC50 = 4000 nM T79031 CO9M2I 46881524 IC50 = 10100 nM T79031 CXG1J4 46881525 IC50 = 22400 nM T79031 CK2SX4 46881526 IC50 = 70500 nM T79031 CC0V6G 46881567 IC50 = 370 nM T79031 C96UFO 46881570 IC50 > 100000 nM T79031 CZ9F5K 46881571 IC50 > 100000 nM T79031 C18ZJA 46881572 IC50 > 100000 nM T79031 C2A9IO 46881612 IC50 > 100000 nM T79031 CCQ5D1 46881613 IC50 = 1710 nM T79031 CO5QC2 46881646 IC50 = 2700 nM T79031 C7C2EK 46881691 IC50 = 4200 nM T79031 CWB9C6 46881692 IC50 = 580 nM T79031 CJN4Y2 46881693 IC50 = 25 nM T79031 CZMJ65 46881696 IC50 = 310 nM T79031 C92QLM 46881697 IC50 = 18100 nM T79031 C5LB4P 46881749 IC50 = 5720 nM T79031 C5G8ZM 46881795 IC50 = 5 nM T79031 CJ3L2B 46881837 IC50 = 16300 nM T79031 CS0O9T 46883935 IC50 = 39.99 nM T79031 CDO30L 46883936 IC50 = 3810 nM T79031 C7O3XP 46884002 IC50 = 29.99 nM T79031 C0GZ5N 46884524 IC50 = 810 nM T79031 C4UOK5 46884581 IC50 = 290 nM T79031 CH42JI 46884664 IC50 = 70 nM T79031 C5N0CB 46887296 Ki = 31 nM T79031 C8NCS9 46887297 Ki = 186 nM T79031 CLO9X6 46887344 Ki = 8 nM T79031 CBIC72 46887345 Ki = 17 nM T79031 CS97BG 46887346 Ki = 22 nM T79031 CZ8XM0 46887347 Ki = 20 nM T79031 CD9AU3 46887394 Ki = 8 nM T79031 C52MSN 46887395 Ki = 12 nM T79031 CHNL31 46887636 IC50 = 10.2 nM T79031 CG10XN 46887637 IC50 = 10.6 nM T79031 C3U9RW 46888932 Ki = 5 nM T79031 CL15AW 46888933 Ki = 60 nM T79031 CZ9NU1 46888934 Ki = 400 nM T79031 CZ6V0R 46888935 Ki = 7 nM T79031 CRW98A 46888936 Ki = 42 nM T79031 C5VNE0 46888937 Ki = 20 nM T79031 CBO5I4 46888938 Ki = 120 nM T79031 CWJ96N 46888939 Ki = 310 nM T79031 CE0L9I 46888940 Ki = 73 nM T79031 C79HMD 46888941 Ki = 45 nM T79031 CU53SL 46888942 Ki = 3 nM T79031 CVP62R 46888943 Ki = 7 nM T79031 CKG8F1 46888944 Ki = 8 nM T79031 C8E6IB 46888945 Ki = 10 nM T79031 CD7GY5 46888946 Ki = 53 nM T79031 CH89KD 46888947 Ki = 240 nM T79031 CWT7E5 46888948 Ki = 970 nM T79031 C1X3MN 46888949 Ki = 1200 nM T79031 C4QJ2C 46888950 Ki = 5800 nM T79031 CV1AN4 46888951 Ki = 73 nM T79031 C36XLK 46888952 Ki = 95 nM T79031 C07TZK 46888953 Ki = 3 nM T79031 CJI24V 46888954 Ki = 1 nM T79031 CIGY12 46888955 Ki = 1 nM T79031 CIH5N4 46888956 Ki = 1 nM T79031 C3MU4T 46888957 Ki = 14 nM T79031 C7O8YN 46888958 Ki = 365 nM T79031 C65CLO 46888959 Ki = 1 nM T79031 CFH1K7 46888960 Ki = 2 nM T79031 C75DZR 46888961 Ki = 1 nM T79031 CF61SW 46888962 Ki = 2 nM T79031 CO7JH5 46888963 Ki = 7 nM T79031 CT1IV9 46888964 Ki = 13 nM T79031 CIG8O7 46888965 IC50 = 490 nM T79031 C76UEW 46891887 IC50 = 470 nM T79031 CK19TM 46893204 IC50 = 4000 nM T79031 CM9IB4 46906639 IC50 = 100000 nM T79031 CH02VP 46906682 IC50 = 11900 nM T79031 CB95GT 46906685 IC50 = 500000 nM T79031 CK34MU 46906686 IC50 = 50000 nM T79031 C2HW5N 46906726 IC50 = 500000 nM T79031 C07OXA 46906809 IC50 = 1000 nM T79031 CLZ7A0 46906811 IC50 = 3700 nM T79031 CGM3Z7 46906869 IC50 = 500000 nM T79031 CI8X9Q 46906870 IC50 = 25000 nM T79031 C4F0RM 46906871 IC50 = 13000 nM T79031 C4V6JC 46906879 IC50 = 30200 nM T79031 C7BTY6 46906915 IC50 = 1900 nM T79031 C5TC1P 46906917 IC50 = 44700 nM T79031 C80RQU 46906956 IC50 = 4000 nM T79031 CKB75W 46906960 IC50 = 12000 nM T79031 C0Z5WQ 46906988 IC50 = 500000 nM T79031 C3VR1T 46906993 IC50 = 2200 nM T79031 C84BKF 46907048 IC50 = 100000 nM T79031 CAP7J3 46907116 IC50 = 100000 nM T79031 CYU07C 46907117 IC50 = 100000 nM T79031 CR2UD5 46907194 IC50 = 100000 nM T79031 C5ZU3L 46907450 IC50 = 16200 nM T79031 CT60JK 46907451 IC50 = 14900 nM T79031 CT47KP 46907452 IC50 = 9500 nM T79031 CT91HV 46907453 IC50 = 8100 nM T79031 CKN35P 46907454 IC50 = 11000 nM T79031 CEUF10 46907455 IC50 = 21400 nM T79031 C70RFN 46907456 IC50 = 15200 nM T79031 CW30MN 46907457 IC50 = 15500 nM T79031 CCS9V5 46907458 IC50 = 9000 nM T79031 C8QTM4 46907484 IC50 = 32800 nM T79031 CV1X4M 46907485 IC50 = 29600 nM T79031 CTF14I 46907486 IC50 = 31200 nM T79031 C4M7IZ 46907487 IC50 = 5 nM T79031 CVN1C5 46911278 IC50 = 350 nM T79031 CY36NG 46927945 IC50 = 88 nM T79031 CY7ZW5 46937311 IC50 = 2770 nM T79031 C0WPX2 46938754 IC50 = 1200 nM T79031 CHT53N 49797544 IC50 = 3 nM T79031 CD4W0Y 49797545 IC50 = 69 nM T79031 C9PRQ0 49800141 IC50 = 10310 nM T79031 CBW81T 49800161 IC50 = 139 nM T79031 C2L0JP 49817351 IC50 = 190 nM T79031 CV86KN 49819085 IC50 = 1 nM T79031 CTP13K 49831178 IC50 = 230 nM T79031 CI8FT3 49836033 IC50 = 12 nM T79031 C65YMH 49855492 IC50 = 270 nM T79031 C12FKR 49855495 IC50 = 330 nM T79031 CP3M8H 49855496 IC50 = 32 nM T79031 CKT38C 49855683 IC50 = 400 nM T79031 C8KA3J 49855886 IC50 = 97 nM T79031 CN7YU1 49858374 IC50 = 1300 nM T79031 CT7H1S 49858375 IC50 = 170 nM T79031 CW9NX3 49858377 IC50 = 490 nM T79031 C3ZON0 49862037 IC50 = 380 nM T79031 CQTW34 49862038 IC50 = 130 nM T79031 C2QIG4 49862039 IC50 = 410 nM T79031 CR0B4M 49862076 IC50 = 166 nM T79031 CD1OV3 49862077 IC50 = 6200 nM T79031 CYT5V1 49862078 IC50 = 260 nM T79031 C79RZN 49862079 IC50 = 720 nM T79031 CBZ7U1 49862117 IC50 = 1100 nM T79031 C6X1YB 49862118 IC50 = 120 nM T79031 CT7HJ8 49862159 IC50 = 370 nM T79031 CHO8L5 49862160 IC50 = 110 nM T79031 C7TH3N 49862161 IC50 = 1600 nM T79031 CPDY93 49862162 IC50 = 7700 nM T79031 C5LAR7 49862202 IC50 = 940 nM T79031 C2EX5O 49862203 IC50 = 180 nM T79031 CO8Q6E 49862204 IC50 = 820 nM T79031 C2IX1G 49862243 IC50 = 1300 nM T79031 CPL1A8 49862244 IC50 = 1400 nM T79031 C09JFC 49862245 IC50 = 800 nM T79031 C3NP6F 49862246 IC50 > 10000 nM T79031 C4YTJ8 49862291 IC50 = 340 nM T79031 C8QO1Y 49862292 IC50 = 250 nM T79031 CDMS96 49862293 IC50 = 1300 nM T79031 CI5HA9 49862343 IC50 = 1000 nM T79031 C5Q3WH 49862344 IC50 = 750 nM T79031 C8BKR7 49862345 IC50 = 560 nM T79031 CVC86Q 49862408 IC50 = 700 nM T79031 C0HEC9 49862409 IC50 = 580 nM T79031 CG36PW 49862410 IC50 = 580 nM T79031 C4YB6V 49862411 IC50 = 1700 nM T79031 CNK03A 49862453 IC50 = 4000 nM T79031 CYFV71 49862454 IC50 = 2400 nM T79031 CV6O8K 49862455 IC50 = 1900 nM T79031 CIH6C5 49862829 IC50 = 460 nM T79031 CKQP37 49862830 IC50 > 10000 nM T79031 C12RTI 49862831 IC50 = 100 nM T79031 CR41SW 49863021 IC50 = 6300 nM T79031 C9O7UP 49863022 IC50 = 1300 nM T79031 C9OWG2 49863023 IC50 = 300 nM T79031 CNC25U 49863024 IC50 = 180 nM T79031 CED4S9 49863025 IC50 = 7900 nM T79031 CCY4G0 49863026 IC50 = 5500 nM T79031 C8T0LZ 49863027 IC50 = 13000 nM T79031 CSYU53 49863028 IC50 = 44000 nM T79031 C64OTC 49863029 IC50 = 50000 nM T79031 CWP2N9 49863030 IC50 = 41000 nM T79031 CWK1B5 49863031 IC50 = 910 nM T79031 CFEP48 49863788 IC50 > 44250 nM T79031 CH1ID2 49863789 IC50 > 42820 nM T79031 C15IFB 49863804 IC50 = 29400 nM T79031 CA45LD 49863805 IC50 > 42460 nM T79031 CL8ZJ9 49863806 IC50 = 37630 nM T79031 C5UEK7 49863807 IC50 = 27850 nM T79031 C64MFI 49863808 IC50 > 45250 nM T79031 C0JRD5 49864293 IC50 = 235000 nM T79031 CMDF79 49864294 IC50 = 54000 nM T79031 C2PMA7 49864484 IC50 = 1008000 nM T79031 CI31WK 49864505 IC50 = 1403000 nM T79031 C2MKA7 49864506 IC50 = 193000 nM T79031 C0U3JM 49864507 IC50 = 827000 nM T79031 CK08EC 49864531 IC50 = 444000 nM T79031 C5C3ZD 49864532 IC50 = 426000 nM T79031 CH2RB1 49864533 IC50 = 83000 nM T79031 CH14WK 49864534 IC50 = 325000 nM T79031 C1ACD7 49864535 IC50 = 249000 nM T79031 CGF02P 49864536 IC50 = 2854000 nM T79031 CWH92P 49864603 IC50 = 194000 nM T79031 C3U8JN 49864604 IC50 = 59000 nM T79031 C2TU5M 49864605 IC50 = 516000 nM T79031 C9OT1N 49864606 IC50 = 72000 nM T79031 C5Y6RD 49864607 IC50 > 1000000 nM T79031 C7ES1O 49864667 IC50 = 246000 nM T79031 CO7X0E 49864668 IC50 = 695000 nM T79031 CN98ZU 49864669 IC50 = 440000 nM T79031 CB5UH7 49864670 IC50 = 243000 nM T79031 CRT6U8 49864671 IC50 = 270000 nM T79031 C21PQB 49864691 IC50 = 375000 nM T79031 CNF53X 49864692 IC50 > 1000000 nM T79031 CV4UF0 49864693 IC50 > 1000000 nM T79031 CX56WY 49864694 IC50 = 8900 nM T79031 CTZR78 49864695 IC50 = 95000 nM T79031 C0MN7Z 49864725 IC50 = 340000 nM T79031 C61YVZ 49864726 IC50 = 264000 nM T79031 C4VM1L 49864727 IC50 = 168000 nM T79031 CC0UO9 49864728 IC50 = 75000 nM T79031 CDX06E 49864729 IC50 = 87000 nM T79031 C8AJ5K 49869035 IC50 = 2200 nM T79031 C1WM9N 49869037 IC50 = 4300 nM T79031 CAPI06 49869040 IC50 = 660 nM T79031 CG5IV6 49869041 IC50 = 4000 nM T79031 C1WYF9 49869172 IC50 = 1700 nM T79031 CR0D3P 49869174 IC50 = 710 nM T79031 C19EDA 49869312 IC50 = 310 nM T79031 CD62TH 49869313 IC50 = 79 nM T79031 CMB32F 49869877 IC50 = 58 nM T79031 CC8O6E 49870864 IC50 = 2300 nM T79031 CB6K7Y 49870865 IC50 = 1900 nM T79031 CVD2Q3 50898620 IC50 = 1490 nM T79031 CO3CN1 50898731 IC50 = 11.9 nM T79031 CVL78S 50904994 IC50 = 45 nM T79031 CBK0C4 50912806 IC50 = 92 nM T79031 CI2VH7 50912937 IC50 = 300 nM T79031 CQK57S 50913659 IC50 = 17 nM T79031 C63QYC 50914101 IC50 = 240 nM T79031 C3A4DL 50914255 IC50 = 4 nM T79031 C29LCP 50914398 IC50 = 30 nM T79031 CJV89L 50914546 IC50 = 8 nM T79031 CTC62N 50914981 IC50 = 32 nM T79031 C92SGN 50937466 IC50 = 150 nM T79031 C5YCV3 50991508 IC50 = 3 nM T79031 CQ31VZ 50991585 IC50 = 9.1 nM T79031 CTL9U5 50991953 IC50 = 120 nM T79031 CA43KF 51026481 IC50 > 5000 nM T79031 CD64NT 51039270 IC50 < 0.54 nM T79031 C0KE4A 52918159 IC50 = 6520 nM T79031 CK1E3W 52918160 IC50 = 11210 nM T79031 CJ6M8H 52940810 EC50 = 220 nM T79031 C3DN8M 52940827 IC50 = 30 nM T79031 CI6H8S 52940883 EC50 = 3140 nM T79031 CVT4K3 52940915 EC50 = 810 nM T79031 CK6N5C 52940942 EC50 = 30 nM T79031 C4DM7B 52940973 EC50 = 270 nM T79031 CD4JE0 52940974 EC50 = 40 nM T79031 CKS25O 52941021 EC50 = 530 nM T79031 C51BHO 52941030 EC50 = 90 nM T79031 CH9ML5 52941133 IC50 = 6900 nM T79031 CLM4T9 52941346 IC50 = 341 nM T79031 C5ZAD4 52941347 IC50 = 640 nM T79031 C5M2TI 52941360 IC50 = 4010 nM T79031 CD4Y3W 52941431 IC50 = 320 nM T79031 CI4RQ0 52941475 IC50 = 131 nM T79031 CJPM97 52941677 EC50 = 70 nM T79031 CZ9ME6 52942030 EC50 = 4320 nM T79031 CLJ01Q 52942108 IC50 = 10 nM T79031 CKU60L 52942135 IC50 = 290 nM T79031 CJ8ZW4 52942210 IC50 = 110 nM T79031 CL56KH 52942211 EC50 = 270 nM T79031 CG24ID 52942212 IC50 = 200 nM T79031 CAOU31 52942213 IC50 = 760 nM T79031 CI35TS 52942269 IC50 = 5400 nM T79031 C4G9QN 52942282 IC50 = 290 nM T79031 CX16LC 52942291 IC50 = 1240 nM T79031 C5K0EN 52942331 IC50 = 5100 nM T79031 CI8CX5 52942524 IC50 = 140 nM T79031 CEJ80Q 52942712 IC50 = 104 nM T79031 CVG51P 52942779 IC50 = 137800 nM T79031 CHN91J 52942848 IC50 = 22 nM T79031 CUZ6X8 52943269 EC50 = 100 nM T79031 CRQ53J 52943292 EC50 = 130 nM T79031 C4LT5U 52943302 EC50 = 20 nM T79031 C60CXD 52943333 EC50 = 120 nM T79031 CS4L9X 52943334 EC50 = 50 nM T79031 C75JQP 52943337 IC50 = 1700 nM T79031 C4TO3K 52943373 EC50 = 100 nM T79031 C4DWX6 52943931 IC50 = 4457 nM T79031 C5QA0I 52943965 IC50 = 1580 nM T79031 CFX8M2 52944038 IC50 = 180 nM T79031 C9MLZ6 52944049 IC50 = 210 nM T79031 C7J3ZR 52944055 IC50 = 1300 nM T79031 CO83YP 52944109 EC50 = 90 nM T79031 C56XOV 52944411 EC50 = 330 nM T79031 CQPD40 52944421 EC50 = 10 nM T79031 CPL95U 52944532 EC50 = 40 nM T79031 C79PAB 52944662 IC50 = 4700 nM T79031 CNQ5Y9 52944681 IC50 = 20 nM T79031 CZ46SX 52944682 IC50 = 10 nM T79031 C4PVH3 52944685 IC50 = 200 nM T79031 C8B2TR 52944893 IC50 = 392 nM T79031 C7W3MN 52945011 IC50 = 720 nM T79031 CJL20O 52945191 IC50 = 1840 nM T79031 CB3QK9 52945497 IC50 = 17200 nM T79031 C58HOG 52945584 IC50 = 4900 nM T79031 C0JQT1 52945785 IC50 = 610 nM T79031 CB9OC2 52945793 EC50 = 5370 nM T79031 CP4WO3 52945841 IC50 = 160 nM T79031 CQ4V8R 52946545 IC50 = 70 nM T79031 C4QLW2 52946836 IC50 = 318 nM T79031 C6D8PN 52946837 IC50 = 3050 nM T79031 CO16KF 52946886 IC50 = 346 nM T79031 CIM9B8 52946887 IC50 = 870 nM T79031 CH8U9I 52946915 IC50 = 50 nM T79031 CRIQ87 52946950 EC50 = 370 nM T79031 CWC0D6 52946966 EC50 = 320 nM T79031 CK2TW7 52947058 IC50 = 6900 nM T79031 CG8AI7 52947059 IC50 = 450 nM T79031 CRNL23 52947103 EC50 = 400 nM T79031 CQ73NP 52947109 EC50 = 100 nM T79031 CAYH50 52947147 EC50 = 1120 nM T79031 CAL2H1 52947347 IC50 = 154 nM T79031 C5UV2T 52947441 IC50 = 30000 nM T79031 C43VCX 52947515 IC50 = 223 nM T79031 C45HZM 52948018 IC50 = 77 nM T79031 C6IC7P 52948105 IC50 = 93 nM T79031 CB3NQ0 52948140 IC50 = 32 nM T79031 C0EPQ2 52948146 EC50 = 80 nM T79031 CY34UI 52948154 EC50 = 70 nM T79031 CKT0J6 52948174 EC50 = 10 nM T79031 CN9H1C 52948200 IC50 = 90 nM T79031 C3N2IQ 52948201 EC50 = 300 nM T79031 CX4JT5 52948286 IC50 = 980 nM T79031 CHIL29 52948341 IC50 = 110 nM T79031 C41NBE 52948410 IC50 = 6300 nM T79031 C4PM0H 52948413 IC50 = 5400 nM T79031 C9QI2S 52948682 IC50 = 46 nM T79031 C8YOD0 52948683 IC50 = 780 nM T79031 CQS24C 52948726 IC50 = 174 nM T79031 CPR34K 52948727 IC50 = 1620 nM T79031 C15VEP 52948732 IC50 = 352 nM T79031 CZ0DX7 52949259 IC50 = 42880 nM T79031 CIT74G 52949295 IC50 = 170 nM T79031 C12DGV 52949296 IC50 = 9360 nM T79031 C51IEW 52949415 IC50 > 50000 nM T79031 CAGS10 52949452 IC50 = 1300 nM T79031 CE27DF 52949464 IC50 = 20 nM T79031 C97IMR 52949465 EC50 = 60 nM T79031 C2XIY3 52949466 IC50 = 20 nM T79031 C5O9AP 52949507 IC50 = 390 nM T79031 CM30YD 52949543 EC50 = 150 nM T79031 CA56UD 52949889 IC50 = 2100 nM T79031 CM7A0X 52949992 IC50 = 4316 nM T79031 C25NMI 52949993 IC50 = 1740 nM T79031 CPO5A7 52950127 EC50 = 50 nM T79031 CKQ34B 52950166 IC50 = 2400 nM T79031 CJ2FB6 52950209 EC50 = 40 nM T79031 CH1T0J 52951738 IC50 = 45.5 nM T79031 C2D1JV 53230332 IC50 = 16 nM T79031 C39RGN 53235196 IC50 = 83 nM T79031 CE3D0S 53236890 IC50 = 74 nM T79031 C1TL7J 53237109 IC50 = 3.7 nM T79031 CI6NF1 53237781 IC50 = 31 nM T79031 C32QSO 53240812 IC50 = 42 nM T79031 C8RV1B 53241150 IC50 = 1 nM T79031 C6V5GK 53241151 IC50 = 10 nM T79031 C17AMV 53241205 IC50 = 110 nM T79031 CLZC60 53241206 IC50 = 17 nM T79031 CDQJ08 53241302 IC50 = 13 nM T79031 CJ24DQ 53241445 IC50 = 3.7 nM T79031 CA9EF1 53241709 IC50 = 17 nM T79031 CC86WU 53241710 IC50 = 13 nM T79031 CR2AW3 53241825 IC50 = 13 nM T79031 C0BRK7 53241826 IC50 = 230 nM T79031 CZ56VB 53241932 IC50 = 23 nM T79031 C7H1ZP 53241933 IC50 = 108 nM T79031 C2F8QG 53241937 IC50 = 131 nM T79031 C6HG0N 53252201 IC50 = 4.4 nM T79031 C6J7UI 53262012 IC50 = 25 nM T79031 CI21EZ 53307133 IC50 = 7000 nM T79031 CMKI49 53307134 IC50 = 2000 nM T79031 C4R8TA 53316808 IC50 = 430 nM T79031 CV9XT5 53316829 IC50 > 10000 nM T79031 CI4RG6 53316830 IC50 = 3000 nM T79031 C3DIM5 53316912 IC50 = 1900 nM T79031 CF2DY9 53317688 IC50 > 10000 nM T79031 C8R5FY 53318147 IC50 > 10000 nM T79031 CQA2R7 53318217 IC50 = 240 nM T79031 C6Y5VL 53319489 IC50 > 10000 nM T79031 CDL09O 53320785 IC50 = 680 nM T79031 CHC91A 53320786 IC50 > 10000 nM T79031 C1WJ0O 53320787 IC50 > 10000 nM T79031 CI4O5J 53320863 IC50 = 50 nM T79031 C8TG1H 53321657 IC50 > 10000 nM T79031 C7NAZ6 53322060 IC50 = 400 nM T79031 CV6K8W 53322096 IC50 > 10000 nM T79031 CJV56W 53322097 IC50 > 10000 nM T79031 C1N2TP 53322098 IC50 > 10000 nM T79031 C0HTX3 53322099 IC50 = 440 nM T79031 CZYC57 53322100 IC50 > 10000 nM T79031 C6ZFR3 53322101 IC50 = 4400 nM T79031 C5AZH3 53322198 IC50 = 3700 nM T79031 CWUZ14 53322199 IC50 > 10000 nM T79031 CFCZ16 53323445 IC50 = 870 nM T79031 CZ72KP 53323446 IC50 > 10000 nM T79031 CQMG75 53323447 IC50 = 6100 nM T79031 CN0PW3 53323448 IC50 > 10000 nM T79031 C8YN6A 53324740 IC50 = 1400 nM T79031 C8KZT6 53324766 IC50 > 10000 nM T79031 CQIX02 53324767 IC50 > 10000 nM T79031 C3DL8J 53324768 IC50 > 10000 nM T79031 C9O2CI 53324843 IC50 > 10000 nM T79031 CM3OP0 53325758 IC50 = 20 nM T79031 C61FYW 53326116 IC50 = 3100 nM T79031 CXY4G5 53326117 IC50 > 10000 nM T79031 C7X1SC 53346491 IC50 = 18 nM T79031 C89HDA 53346495 IC50 = 30902.95 nM T79031 CHJ6X1 53379400 IC50 = 11.6 nM T79031 C1QYU2 53464257 IC50 = 0.2 nM T79031 C6KC5V 53464567 IC50 = 0.2 nM T79031 C4Q0JV 53464571 IC50 = 0.3 nM T79031 CPE0Q3 53464695 IC50 = 1.2 nM T79031 CG7NH3 53464819 IC50 = 12 nM T79031 CC7P2U 53464882 IC50 = 19 nM T79031 CPRZ03 53464941 IC50 = 2.7 nM T79031 CRA3L0 53464942 IC50 = 3 nM T79031 CYE6O4 53464943 IC50 = 2.6 nM T79031 C3I8KD 53464944 IC50 = 0.3 nM T79031 C6K5JY 53464945 IC50 = 0.7 nM T79031 CK8YI4 53465003 IC50 = 5 nM T79031 C9K6FT 53465005 IC50 = 7 nM T79031 CH9CX8 53465067 IC50 = 0.5 nM T79031 CRW3C5 53465113 IC50 = 0.3 nM T79031 C17GML 53465141 IC50 = 3 nM T79031 CVM91G 53465142 IC50 = 0.4 nM T79031 C6H0YB 53465848 IC50 = 5200 nM T79031 CBE4M7 53465849 IC50 = 34 nM T79031 CD5O2N 53465850 IC50 = 2.5 nM T79031 C3FW4L 53465851 IC50 = 970 nM T79031 CL50RP 53465913 IC50 = 16 nM T79031 CFV4D5 53465914 IC50 = 27 nM T79031 CO4UL9 53465915 IC50 = 11 nM T79031 CVO9T7 53465916 IC50 = 0.65 nM T79031 CIC97W 53465917 IC50 = 20 nM T79031 CF6ED5 53465918 IC50 = 88 nM T79031 C1S5JT 53465989 IC50 = 50 nM T79031 C3I0EQ 53465990 IC50 = 10 nM T79031 CN2G8B 53465991 IC50 = 16 nM T79031 CQ76IP 53465992 IC50 = 80 nM T79031 CQ80DR 53465993 IC50 = 97 nM T79031 CL3ZV6 53466061 IC50 = 390 nM T79031 CS27FE 53466062 IC50 = 15 nM T79031 CU9R8S 53481984 IC50 = 36 nM T79031 C7Z9TI 53484158 IC50 = 270 nM T79031 C2RU1J 53493350 EC50 = 17 nM T79031 C17NYM 53493353 EC50 = 9 nM T79031 CZ7UV6 53493354 EC50 = 53 nM T79031 C86VQT 53494150 EC50 = 317 nM T79031 C2GUC3 53494692 EC50 = 16 nM T79031 C1T6KF 53494828 EC50 = 1884 nM T79031 C2GC5Y 54577358 IC50 = 11 nM T79031 CUSF85 54577394 IC50 = 1000 nM T79031 CXOH83 54577607 IC50 = 400 nM T79031 C5OP2B 54577822 IC50 = 1 nM T79031 C8SJA4 54578013 IC50 = 142000 nM T79031 CF40KI 54580003 IC50 = 4570 nM T79031 C6N0JA 54580022 IC50 = 11150 nM T79031 CXF10V 54580145 IC50 = 1200 nM T79031 CF80UT 54581101 IC50 = 55000 nM T79031 C6YPJ3 54581139 IC50 > 100000 nM T79031 CFM91Y 54581140 IC50 = 4200 nM T79031 C1FSR5 54582051 IC50 = 9100 nM T79031 CHT6G1 54582052 IC50 = 12120 nM T79031 CEID56 54583000 IC50 = 23920 nM T79031 C3ROW7 54583129 IC50 = 6200 nM T79031 CB41FM 54583130 IC50 = 550 nM T79031 CM5H4C 54583965 IC50 = 8980 nM T79031 CO6T7C 54584085 IC50 = 1100 nM T79031 C8UN3G 54584123 IC50 = 4300 nM T79031 C6C2NO 54585055 IC50 = 60 nM T79031 CX47YB 54585056 IC50 = 66000 nM T79031 C8G1UV 54585911 IC50 = 11290 nM T79031 C7KU6J 54586032 IC50 = 3200 nM T79031 CY58NP 54586033 IC50 = 1400 nM T79031 CJ2RN8 54587663 IC50 = 103500 nM T79031 C8DL4Y 54729809 IC50 = 100000 nM T79031 CTR1F7 54760130 IC50 = 1148 nM T79031 C3M8AQ 54760132 IC50 = 348 nM T79031 CT39AH 54760133 IC50 = 1380 nM T79031 CMFA14 54760134 IC50 = 151 nM T79031 C7IYH0 54760314 IC50 > 10000 nM T79031 CTLV61 54761047 IC50 = 710 nM T79031 C80STN 54761221 IC50 = 27.7 nM T79031 C2G0TL 54765328 IC50 = 150 nM T79031 CDRO32 55281242 IC50 = 8200000 nM T79031 CNM1V5 56589875 IC50 = 26 nM T79031 CRV6N7 56593478 IC50 = 23.44 nM T79031 CQ23ZS 56600729 IC50 = 83 nM T79031 CN09BJ 56645128 IC50 = 3 nM T79031 CKM5G6 56657790 IC50 = 130 nM T79031 C2MHC3 56657791 IC50 = 69 nM T79031 CO8MD5 56657792 IC50 = 250 nM T79031 CG1D6V 56658432 EC50 = 490 nM T79031 C0RMT9 56658435 EC50 = 110 nM T79031 C2J7TS 56658436 IC50 = 70 nM T79031 CW8IY4 56658437 EC50 = 2230 nM T79031 C45YJU 56658717 EC50 = 500 nM T79031 CS4MX1 56658718 EC50 = 300 nM T79031 C7JKI8 56661313 IC50 = 250 nM T79031 CX54RO 56661314 IC50 > 91000 nM T79031 CO5X3E 56661417 IC50 = 40.6 nM T79031 CH2A6Q 56661551 IC50 = 39.6 nM T79031 CM4P2G 56661917 IC50 = 30 nM T79031 C4QD7Z 56661918 IC50 = 80 nM T79031 C47HVP 56661919 EC50 = 150 nM T79031 C0FCR2 56663019 IC50 = 2400 nM T79031 CQP28A 56665390 IC50 = 20 nM T79031 CCLI91 56668288 IC50 = 24.8 nM T79031 C2CO7G 56668394 IC50 = 34.8 nM T79031 CZO04V 56668395 IC50 = 31.9 nM T79031 C39XJR 56668818 IC50 = 1960 nM T79031 CXW4B7 56668819 IC50 = 20 nM T79031 C1Z7MG 56668820 EC50 = 370 nM T79031 C10MSR 56668821 EC50 = 10 nM T79031 C5VIR4 56669107 IC50 = 80 nM T79031 C1DFQ6 56672294 IC50 = 70 nM T79031 CFE52J 56672296 EC50 = 1170 nM T79031 C2EZ8O 56672297 EC50 = 500 nM T79031 CGNH26 56672298 IC50 = 15 nM T79031 CCG59L 56672299 EC50 = 200 nM T79031 CLP36K 56672300 EC50 = 220 nM T79031 CL26PC 56675093 IC50 = 140 nM T79031 C1AC2N 56675287 IC50 = 29 nM T79031 C43PXS 56675689 IC50 = 10 nM T79031 CL8PK3 56675694 IC50 = 180 nM T79031 CV3BE8 56675695 EC50 = 450 nM T79031 CUI46G 56675696 EC50 = 30 nM T79031 C08UNH 56678401 IC50 = 180 nM T79031 CP6KX7 56678402 IC50 = 260 nM T79031 CM8R3U 56678616 IC50 = 20.4 nM T79031 CF9P5T 56678617 IC50 = 24.2 nM T79031 CO7G3P 56678998 IC50 = 16 nM T79031 C65LKQ 56678999 IC50 = 370 nM T79031 CLW2C5 56679000 EC50 = 370 nM T79031 C1UO5J 56679223 IC50 = 42 nM T79031 CH80FW 56679262 IC50 = 100 nM T79031 CC5A6E 56680040 IC50 = 3400 nM T79031 CM78OG 56681734 IC50 = 110 nM T79031 CNXQ68 56681735 IC50 = 220 nM T79031 CXJ4Z3 56681789 IC50 = 100000 nM T79031 CD92CR 56681945 IC50 = 27 nM T79031 CGL67Z 56682312 IC50 = 20 nM T79031 C07EXO 56682313 IC50 = 140 nM T79031 CE8PW7 56682314 EC50 = 2900 nM T79031 C7QB6A 56682567 EC50 = 1700 nM T79031 CBVK48 56834873 Ki = 17 nM T79031 C8MU0G 56834948 IC50 = 24 nM T79031 C7SIV2 56834949 IC50 = 29 nM T79031 C1G6KL 56834950 IC50 = 36 nM T79031 C4KP9I 56925448 Ki = 5312 nM T79031 C0ZKP8 56925449 Ki = 2389 nM T79031 CQE1L7 56925450 Ki = 2160 nM T79031 C9DH8A 56925452 Ki = 495 nM T79031 CMSO49 56925453 Ki = 301 nM T79031 CG3C2H 56925544 IC50 = 178 nM T79031 CE9YN7 56925547 Ki = 926 nM T79031 C92CRT 56925548 Ki = 34 nM T79031 CNV7I5 56925549 Ki = 25 nM T79031 CI2KX3 56928834 IC50 = 60 nM T79031 C2H7BK 56935646 IC50 = 3800 nM T79031 CT2LF3 56935647 IC50 = 2500 nM T79031 C2HT1W 56935716 IC50 = 700 nM T79031 CF76QP 56940703 IC50 = 1100000 nM T79031 C40GTY 56940704 IC50 = 242000 nM T79031 C9F3MT 56940705 IC50 = 114000 nM T79031 CMDN82 56940706 IC50 = 33000 nM T79031 CNC1D9 56940707 IC50 = 7000 nM T79031 C8HW0J 56940710 IC50 = 11000 nM T79031 CZ38BR 56940711 IC50 = 6260 nM T79031 C9KI7Q 56940718 IC50 = 18 nM T79031 CGZ0M9 56944167 IC50 = 4930 nM T79031 CH8FO4 56947420 IC50 = 21 nM T79031 C4ZSQ1 56947421 IC50 = 5.4 nM T79031 CP2DE0 56947553 IC50 = 7.3 nM T79031 C6BW5Q 56947557 IC50 = 11 nM T79031 C4K1XS 56947558 IC50 = 28 nM T79031 C0NH9E 56947697 IC50 = 16 nM T79031 CT2M3V 56947698 IC50 = 26 nM T79031 CZ4M0T 56947699 IC50 = 27 nM T79031 C7RZ0B 56947700 IC50 = 21 nM T79031 COHF14 56947701 IC50 = 39 nM T79031 CT0PC4 56947827 IC50 = 5.7 nM T79031 C0KY3J 56947828 IC50 = 19 nM T79031 C63PVB 56947829 IC50 = 61 nM T79031 CA9LP1 56948072 IC50 = 12 nM T79031 CX3E4B 56948453 IC50 = 490 nM T79031 CZ67RX 56948455 IC50 = 670 nM T79031 CPI2Y4 56948542 IC50 = 48.98 nM T79031 C1TG8P 56948806 IC50 = 31 nM T79031 CMA7L0 56954888 IC50 = 22400 nM T79031 C8XCI0 56954891 IC50 = 14400 nM T79031 CHV8U3 56954986 IC50 = 2100 nM T79031 C0JCZ2 56954989 IC50 = 3000 nM T79031 CC7Y5O 56955099 IC50 = 2800 nM T79031 C9XO0M 56955109 IC50 = 2900 nM T79031 COE65B 56955111 IC50 = 3600 nM T79031 C2M6DQ 56955293 IC50 = 13600 nM T79031 C2BUR9 56956281 IC50 = 2 nM T79031 CO2JR1 56969382 IC50 = 54 nM T79031 C3M0IY 57327926 IC50 = 7400 nM T79031 CNIH09 57327927 IC50 = 7320 nM T79031 CL3FK5 57327997 IC50 = 5590 nM T79031 C87FEL 57327999 IC50 = 5950 nM T79031 C7WLS6 57328246 IC50 = 7.943 nM T79031 C0MGN1 57345931 IC50 = 260 nM T79031 CB4DM7 57345932 IC50 = 78 nM T79031 C4BD2H 57384014 IC50 = 86 nM T79031 CMY58P 57384015 IC50 = 82 nM T79031 CP0Z2F 57384016 IC50 = 169 nM T79031 C76CME 57384020 IC50 = 138 nM T79031 C9Q4VL 57384270 IC50 = 2 nM T79031 CDS03B 57384271 IC50 = 210 nM T79031 CBKI24 57384272 IC50 = 950 nM T79031 C6IAW5 57384273 IC50 = 36 nM T79031 C42JEK 57384274 IC50 = 7 nM T79031 C1T0NE 57385371 IC50 = 0.72 nM T79031 C7DI1C 57385528 IC50 = 550 nM T79031 CAR38J 57385530 IC50 = 1360 nM T79031 C90GLN 57385533 IC50 = 1650 nM T79031 C8EYC2 57385625 IC50 = 4.6 nM T79031 CGPA23 57385772 IC50 = 3520 nM T79031 CU9FY0 57385773 IC50 = 2010 nM T79031 C57IRM 57385877 IC50 = 0.56 nM T79031 CA0X8R 57386049 IC50 = 94 nM T79031 CLIW35 57386302 IC50 = 130 nM T79031 C5CF8I 57386304 IC50 = 670 nM T79031 CNAI80 57386563 IC50 = 350 nM T79031 CB4WO2 57386811 IC50 = 55 nM T79031 C5VQE6 57386812 IC50 = 140 nM T79031 COL2R0 57386813 IC50 = 1370 nM T79031 CZT37N 57386814 IC50 = 130 nM T79031 C0TOR5 57387067 IC50 = 55 nM T79031 CG2R8K 57387068 IC50 = 120 nM T79031 C1K6GV 57387069 IC50 = 740 nM T79031 CI7LG6 57387070 IC50 = 140 nM T79031 C07BNE 57387166 IC50 = 2.3 nM T79031 C52VTC 57387317 IC50 = 80 nM T79031 CU3C7S 57387318 IC50 = 115 nM T79031 C2HV9X 57387319 IC50 = 310 nM T79031 C46BLJ 57387320 IC50 = 79 nM T79031 C67AEU 57387579 IC50 = 150 nM T79031 C7ZHD4 57387580 IC50 = 1770 nM T79031 CSC27H 57387581 IC50 = 8 nM T79031 CD36BM 57387582 IC50 = 24 nM T79031 CB5V0D 57387583 IC50 = 120 nM T79031 C5QXU9 57387806 IC50 = 225 nM T79031 CFD9V5 57387807 IC50 = 116 nM T79031 C9DEX6 57387808 IC50 = 75 nM T79031 CZ0W8T 57387809 IC50 = 2 nM T79031 CWLJ62 57387810 IC50 = 43 nM T79031 C3MNK4 57388037 IC50 = 3 nM T79031 CYL8B2 57388039 IC50 > 10000 nM T79031 CP9V7X 57388040 IC50 > 10000 nM T79031 CJA0T7 57388041 IC50 = 68 nM T79031 CIXH43 57388118 IC50 = 0.59 nM T79031 CO3BA4 57390575 Ki = 62 nM T79031 CO7GP3 57390627 IC50 = 11 nM T79031 CWVU97 57390900 IC50 > 10000 nM T79031 CVD9G0 57390901 IC50 > 10000 nM T79031 CY1CH8 57390902 IC50 > 10000 nM T79031 CZ7W0K 57390903 IC50 > 10000 nM T79031 CG6V3B 57391024 IC50 = 3 nM T79031 C9BQF5 57391072 IC50 = 38 nM T79031 C07LEX 57391075 IC50 = 110 nM T79031 C1YSE6 57391110 IC50 = 14200 nM T79031 CO0AH5 57391182 IC50 = 1.3 nM T79031 C5Q2ET 57392204 IC50 = 45 nM T79031 CZ52BC 57392702 IC50 > 10000 nM T79031 C3S8UP 57392703 IC50 > 10000 nM T79031 C0GL9N 57392821 IC50 > 330 nM T79031 CWV34T 57392861 IC50 = 400 nM T79031 C9GNY6 57392862 IC50 = 4.7 nM T79031 CRSU67 57392936 IC50 = 46 nM T79031 CT2EW6 57392937 IC50 = 67 nM T79031 C8PW6Z 57392956 IC50 = 190 nM T79031 C54CGB 57393109 IC50 = 58.88 nM T79031 C3U2BA 57393960 IC50 = 88 nM T79031 CK7OV2 57393961 IC50 = 140 nM T79031 CV2R0K 57394453 IC50 = 57000 nM T79031 C3AT1L 57394592 IC50 = 160 nM T79031 CVS26H 57394593 IC50 = 1400 nM T79031 CLQA20 57394700 IC50 = 330 nM T79031 CVY8I4 57394835 IC50 = 20.42 nM T79031 CRJD62 57394836 IC50 = 12.59 nM T79031 CX2SV8 57394837 IC50 = 13.49 nM T79031 CL9D3P 57395700 IC50 = 15 nM T79031 CQ58OT 57395865 Ki = 304 nM T79031 CVJZ32 57395866 Ki = 180 nM T79031 C1DWL2 57396182 IC50 > 10000 nM T79031 COL67S 57396183 IC50 = 4800 nM T79031 CVC1D5 57396216 IC50 = 240000 nM T79031 C54QAW 57396217 IC50 = 19000 nM T79031 CRF9X0 57396340 IC50 = 4.2 nM T79031 CW8LF9 57396341 IC50 = 2.6 nM T79031 CIDM04 57396342 IC50 = 23 nM T79031 C5EPT1 57396520 IC50 = 3840 nM T79031 C4AW9L 57396605 IC50 = 22.39 nM T79031 CHO31M 57396606 IC50 = 13.8 nM T79031 CO48ZJ 57396607 IC50 = 37.15 nM T79031 C4TNG1 57397484 IC50 = 5 nM T79031 CS81LA 57397485 IC50 = 54 nM T79031 CP87YD 57397486 IC50 = 8 nM T79031 CD5XE6 57397487 IC50 = 17 nM T79031 CMJ4N2 57397488 IC50 = 68 nM T79031 C0JQE1 57397990 IC50 > 10000 nM T79031 CPY29G 57397991 IC50 > 10000 nM T79031 C6UVI3 57398014 IC50 = 600 nM T79031 C19BSQ 57398246 IC50 = 360 nM T79031 CV70IK 57398311 IC50 = 2810 nM T79031 CY5SR1 57399172 IC50 = 1100 nM T79031 C0YAU9 57399319 Ki = 525 nM T79031 CVL27Z 57399320 EC50 = 230 nM T79031 C3DK0O 57399645 IC50 > 10000 nM T79031 C3YQO9 57399646 IC50 = 4700 nM T79031 CI7SL4 57399647 IC50 > 10000 nM T79031 CV93JY 57399788 IC50 = 27 nM T79031 CEW89C 57399789 IC50 = 19 nM T79031 CJ57TR 57399790 IC50 = 55 nM T79031 CJ79QG 57399791 IC50 = 650 nM T79031 CT61PB 57399899 IC50 = 12 nM T79031 C3M7XH 57399972 IC50 = 2270 nM T79031 C3CS7K 57400036 IC50 = 19.5 nM T79031 CZ6KN5 57400037 IC50 = 3388.44 nM T79031 CV3D4S 57400038 IC50 = 34.67 nM T79031 CE7L4P 57400927 IC50 = 141 nM T79031 C02ITG 57400928 IC50 = 600 nM T79031 CR1SG7 57400929 IC50 = 870 nM T79031 CNS8X6 57400930 IC50 = 1200 nM T79031 CA0D5J 57400931 IC50 = 5 nM T79031 C9E8VP 57400932 IC50 = 12 nM T79031 CCW50V 57401070 IC50 = 164.5 nM T79031 C8NEZ3 57401086 Ki = 1041 nM T79031 C25KEQ 57401558 IC50 = 220 nM T79031 C46YGJ 57401559 IC50 = 31 nM T79031 CH6E5J 57401659 IC50 = 220 nM T79031 CJ8B6S 57401671 IC50 = 510 nM T79031 CT58MW 57401672 IC50 = 1.4 nM T79031 C2I7AN 57402628 IC50 = 10 nM T79031 C81RML 57403150 IC50 > 10000 nM T79031 C0R7QC 57403151 IC50 > 10000 nM T79031 CV0EA5 57403152 IC50 > 10000 nM T79031 CU53AZ 57403177 IC50 = 70 nM T79031 C82UVR 57403311 IC50 = 110 nM T79031 C0JF6T 57403385 IC50 = 20 nM T79031 CVTQ25 57403386 IC50 = 210 nM T79031 CRUG76 57403387 IC50 = 5.2 nM T79031 CGPW43 57403388 IC50 = 240 nM T79031 CZI6C7 57403403 IC50 = 40 nM T79031 C3ZPN8 57403404 IC50 = 34 nM T79031 CES1O6 57403718 IC50 > 500000 nM T79031 CJLB64 57404339 Ki = 5.4 nM T79031 C6WU8O 57406717 IC50 = 9.09 nM T79031 C1GEY2 57406719 IC50 = 1.84 nM T79031 C0M6NB 57406720 IC50 = 3.98 nM T79031 CWCY97 57406911 IC50 = 60.8 nM T79031 C62DBF 57407296 IC50 = 5 nM T79031 C1FTY8 57512157 IC50 = 538 nM T79031 C3G2ZX 57515809 IC50 = 31 nM T79031 CC8U3J 57825146 IC50 = 8200 nM T79031 CTU5I7 57825223 IC50 = 5500 nM T79031 CH94PW 57825229 IC50 = 13000 nM T79031 C0PID6 57843652 Ki = 480 nM T79031 CWQ9B4 57844200 Ki = 430 nM T79031 C6WU7P 57844259 Ki = 16 nM T79031 CD9A1M 57844562 Ki = 230 nM T79031 CNJ3G9 57844902 Ki = 3800 nM T79031 CYQ9W6 57855519 IC50 > 2000000 nM T79031 CB81RE 58118813 IC50 = 352 nM T79031 CRBY82 58118864 IC50 = 5 nM T79031 CJZ3Q0 58118873 IC50 = 7 nM T79031 C9FBE0 58118888 IC50 = 28 nM T79031 CD7MY6 58138221 IC50 = 3200 nM T79031 CQUB63 58157954 IC50 = 1800 nM T79031 C0M7QL 58197221 IC50 = 4 nM T79031 CU1FR6 58423762 IC50 = 36830 nM T79031 CZF04E 58443119 Ki = 60 nM T79031 C9OF5W 58443138 Ki = 1463 nM T79031 CI1X9T 58443145 Ki = 783 nM T79031 CC8TK0 58466119 IC50 = 0.9 nM T79031 C9IRW0 58466120 IC50 = 5 nM T79031 CSU91B 58466122 IC50 = 0.7 nM T79031 CKSF73 58466243 IC50 = 0.9 nM T79031 CH9ER4 58466295 IC50 = 6 nM T79031 C6QJX4 58466300 IC50 = 0.6 nM T79031 C6OJC2 58466301 IC50 = 23 nM T79031 C5RXE1 58483782 IC50 = 13700 nM T79031 C0Z8PG 58771867 Ki = 50 nM T79031 C43ZQS 58771881 Ki = 150 nM T79031 CJTL53 58909353 IC50 = 414 nM T79031 C1WF5O 58962911 Ki = 40 nM T79031 CYFB09 58962922 Ki = 860 nM T79031 C6G9WI 58962926 Ki = 2200 nM T79031 C9MQ3C 58962943 Ki = 270 nM T79031 CV29SE 58962956 Ki = 500 nM T79031 C0XK5Q 58962961 Ki = 5 nM T79031 C3VHC7 59028115 IC50 = 45 nM T79031 C9ENH5 59129131 IC50 = 93 nM T79031 C4BOY9 59166662 Ki = 10.8 nM T79031 CAY3S1 59166665 Ki = 63.1 nM T79031 C2K9PU 59250417 IC50 = 7.2 nM T79031 CF20WL 59250968 IC50 = 20 nM T79031 CCS34R 59250998 IC50 = 14 nM T79031 CI2Z1Y 59251000 IC50 = 20 nM T79031 CW63FG 59262280 Ki = 10 nM T79031 CJ54VX 59262314 Ki = 270 nM T79031 C0VJH7 59262316 Ki = 830 nM T79031 CIP54X 59262346 Ki = 860 nM T79031 CFD96H 59262349 Ki = 585 nM T79031 CQO7U1 59262351 Ki = 276 nM T79031 C1Y6QS 59262353 Ki = 3 nM T79031 C78KCH 59262361 Ki = 470 nM T79031 CFJM61 59262417 Ki = 90 nM T79031 CS8KD6 59262423 Ki = 270 nM T79031 CJZ28U 59262424 Ki = 170 nM T79031 CHOY58 59262427 Ki = 470 nM T79031 CDG7K0 59262444 Ki = 110 nM T79031 CEH6P3 59262455 Ki = 88 nM T79031 C5ZIS8 59262464 Ki = 30 nM T79031 C2I0YK 59262465 Ki = 450 nM T79031 CC5J3G 59262483 Ki = 130 nM T79031 CD27WU 59262486 Ki = 350 nM T79031 COXS29 59262510 Ki = 250 nM T79031 CXZ4D2 59262540 Ki = 47 nM T79031 C6Q4EZ 59262553 Ki = 301 nM T79031 CID2C7 59262561 Ki = 10 nM T79031 CHB56R 59262564 Ki = 320 nM T79031 CNAG56 59262582 Ki = 430 nM T79031 C2PJ4N 59271992 IC50 > 30000 nM T79031 C7XM1P 59272333 IC50 = 7 nM T79031 CWCK45 59272335 IC50 = 2 nM T79031 CJKM47 59374702 IC50 = 13 nM T79031 CW9IM6 59374749 IC50 = 22000 nM T79031 C3IT5Q 59387262 Ki = 210 nM T79031 C85IUE 59387407 Ki = 100 nM T79031 CM79PZ 59387534 Ki = 470 nM T79031 C0RCW2 59387607 Ki = 350 nM T79031 CQ85SC 59387748 Ki = 1200 nM T79031 CBH8L1 59388200 Ki = 138 nM T79031 CS9LG6 59388465 Ki = 21 nM T79031 CQ17MD 59388490 Ki = 190 nM T79031 CX28OJ 59388662 Ki = 1200 nM T79031 CPV8T9 59388715 Ki = 1900 nM T79031 CN15RU 59388772 Ki > 10000 nM T79031 CP25LG 60043779 IC50 = 643 nM T79031 CPM5E7 60045607 IC50 < 50000 nM T79031 C6AYV3 60144368 IC50 = 1 nM T79031 CQW7A8 60149247 Ki > 10000 nM T79031 CE7PG1 60164519 IC50 = 7 nM T79031 COXS42 60168050 IC50 = 3 nM T79031 CV43HQ 60168051 IC50 = 5 nM T79031 C60ESV 60194610 IC50 = 2.188 nM T79031 C9E4NW 60202322 IC50 = 5 nM T79031 CG9TQ4 60210990 Ki = 3 nM T79031 CU2IN6 60210991 Ki = 90 nM T79031 CA48QS 62707060 IC50 = 263 nM T79031 CTD1I5 62707061 IC50 = 173 nM T79031 CX4MY0 62707358 IC50 = 163 nM T79031 C3Z7DB 62707359 IC50 = 141 nM T79031 C6I4GR 62707360 IC50 = 184 nM T79031 C6AEZ7 66545742 IC50 = 157000 nM T79031 CKAD71 66545743 IC50 = 4600 nM T79031 CKM38C 66545744 IC50 = 17100 nM T79031 C3V4UC 66549618 IC50 = 142 nM T79031 C6T0AJ 66557874 Ki = 1 nM T79031 CLRC36 66557875 Ki = 6 nM T79031 CLO54N 66557876 Ki = 3 nM T79031 CY3P0N 66558601 IC50 = 1 nM T79031 C0M7FD 66558858 IC50 = 27 nM T79031 CGX98L 66559017 IC50 = 25 nM T79031 C5B6FE 66562362 IC50 = 1 nM T79031 CUE46I 66575069 IC50 = 57.2 nM T79031 CQM8I7 66575075 IC50 = 10 nM T79031 CCN98R 66649578 IC50 = 38 nM T79031 CHS2G5 66649612 IC50 = 124 nM T79031 C75DVR 66649674 IC50 = 32 nM T79031 C2BGY7 66649788 IC50 = 19 nM T79031 CFML30 66665322 IC50 = 10 nM T79031 CB6ZA3 66683197 EC50 = 220 nM T79031 C83LNT 66683198 EC50 = 222 nM T79031 C8N2ZT 66683200 EC50 = 316 nM T79031 CGKU53 66683659 EC50 = 170 nM T79031 CB4WQ9 66683677 IC50 = 32863 nM T79031 C92SYT 66683709 EC50 = 8 nM T79031 CWE7G3 66683751 EC50 = 971 nM T79031 CP09ND 66684067 EC50 = 90 nM T79031 C9AZ1X 66684136 EC50 = 27 nM T79031 C7Z6OV 66684147 EC50 = 8.9 nM T79031 C7X6FL 66684245 EC50 = 896 nM T79031 C1X4GA 66684386 EC50 = 3208 nM T79031 CTW1K5 66930459 IC50 = 7100 nM T79031 C9JG0X 66930522 IC50 = 99300 nM T79031 C86KZM 66930530 IC50 = 270 nM T79031 C35MOD 66930632 IC50 = 2300 nM T79031 C9LQ5R 66930642 IC50 = 1700 nM T79031 CKQ4L1 66930658 IC50 = 3000 nM T79031 CFC10G 66930669 IC50 = 350 nM T79031 CUA98P 66930693 IC50 = 23100 nM T79031 C5T9QN 66930698 IC50 = 5300 nM T79031 CQHC53 66930707 IC50 = 3100 nM T79031 CFT2D8 66930736 IC50 = 1200 nM T79031 CUR61K 66930746 IC50 = 3300 nM T79031 CA83IR 66930761 IC50 = 20900 nM T79031 C0TX7N 66930779 IC50 = 1700 nM T79031 C5U4DI 66930819 IC50 = 6400 nM T79031 CGC47N 67236442 EC50 = 14 nM T79031 C4V3NK 67246237 IC50 = 2470 nM T79031 CM8PJ4 67246553 IC50 = 4540 nM T79031 CYK23N 67246725 IC50 = 2760 nM T79031 CYA5T3 67246787 IC50 = 1170 nM T79031 C7R0IM 67247796 IC50 = 10400 nM T79031 CIT9Y0 67247849 IC50 = 4220 nM T79031 C63VKT 67247971 IC50 = 2230 nM T79031 CV2W4A 67248528 IC50 = 2980 nM T79031 C1DXK4 67248938 IC50 = 800 nM T79031 COGX71 67249135 IC50 = 5060 nM T79031 CEZH46 67269595 IC50 = 9.1 nM T79031 C9W6ER 67269889 IC50 = 5.9 nM T79031 CLU63M 67270136 IC50 = 4.1 nM T79031 CO5FJ0 67270250 IC50 = 28.9 nM T79031 CFNV35 67270281 IC50 = 7.2 nM T79031 C3DY9K 67270599 IC50 = 6.1 nM T79031 CN3OY6 67270633 IC50 = 6.3 nM T79031 CBTS03 67270704 IC50 = 5.5 nM T79031 CK16WC 67270717 IC50 = 9.8 nM T79031 C9AQ0T 67270792 IC50 = 9.8 nM T79031 CVL03S 67270914 IC50 = 9.3 nM T79031 C7QN8E 67270937 IC50 = 5.7 nM T79031 C8EFI1 67270974 IC50 = 12 nM T79031 CI1MQ0 67304745 IC50 = 4 nM T79031 C7DJ6S 67305134 IC50 = 2140 nM T79031 CISX59 67305701 IC50 = 2.4 nM T79031 C5X3ZN 67306893 IC50 = 1.8 nM T79031 CO3ND7 67387844 IC50 = 0.4 nM T79031 CBFE84 67436561 IC50 = 0.3 nM T79031 CUXH49 67463314 IC50 = 1 nM T79031 CHU12R 67950044 IC50 = 20 nM T79031 CU5P3C 67950045 IC50 = 140 nM T79031 CJA86Z 67950104 IC50 = 90 nM T79031 CM9V8X 67950125 IC50 = 39 nM T79031 C7D1ZU 67950129 IC50 = 56 nM T79031 CAK76O 67950143 IC50 = 60 nM T79031 CQ24FC 67950181 IC50 = 35 nM T79031 CEM6I0 67950185 IC50 = 16000 nM T79031 CC4V3N 67950186 IC50 = 76 nM T79031 CC69RG 67950202 IC50 = 23 nM T79031 CDN75Y 67950205 IC50 = 55 nM T79031 C6WS4Z 67950214 IC50 = 150 nM T79031 CDH49P 67950241 IC50 = 130 nM T79031 C2P8SB 67950244 IC50 = 54 nM T79031 CBOC21 67970433 IC50 = 170 nM T79031 C9TXI4 67970604 IC50 = 61 nM T79031 C7KX8J 67970675 IC50 = 400 nM T79031 CH9WP7 67970677 IC50 = 760 nM T79031 C0IG9N 67970973 IC50 = 180 nM T79031 C89UJX 67971074 IC50 = 940 nM T79031 CSK05E 67971135 IC50 = 670 nM T79031 CJ5YT6 67971215 IC50 = 130 nM T79031 C25BUR 67971352 IC50 = 71 nM T79031 C8ZEP9 67971363 IC50 = 830 nM T79031 C2SA9C 67971406 IC50 = 92 nM T79031 CQ93MO 67971614 IC50 = 120 nM T79031 CBO8G1 67971622 IC50 = 17000 nM T79031 C29ONK 67971826 IC50 = 120 nM T79031 CV7BH5 67971878 IC50 = 7700 nM T79031 C8HEF1 67971920 IC50 = 650 nM T79031 CGMR05 67971930 IC50 = 37 nM T79031 C12QLO 67979331 IC50 = 0.72 nM T79031 CDYX41 67979392 IC50 = 1.4 nM T79031 C4V6SP 67979424 IC50 = 1.4 nM T79031 CC8BT6 68111516 Ki = 2.4 nM T79031 CL7R0G 68256677 Ki = 52900 nM T79031 C5QO2U 68256748 Ki = 129 nM T79031 C5XA1S 68307473 IC50 = 52 nM T79031 C7XBG9 68321727 EC50 = 45 nM T79031 C5IP2Z 68321730 IC50 = 39 nM T79031 CLZG95 68321802 IC50 = 28 nM T79031 CN3GX2 68321815 EC50 = 633 nM T79031 C90AYO 68321837 IC50 = 36 nM T79031 CCKG03 68321840 EC50 = 148 nM T79031 CBY7W2 68321854 IC50 = 151 nM T79031 CZM1N6 68321874 EC50 = 399 nM T79031 CGZP43 68321882 IC50 = 68 nM T79031 CVH4Z8 68321895 IC50 = 7197 nM T79031 CT20FH 68321898 IC50 = 2864 nM T79031 CR4W5M 68321900 IC50 = 1701 nM T79031 C9RS4D 68321905 IC50 = 344 nM T79031 C9B5LG 68321915 EC50 = 98 nM T79031 C4LFD5 68321923 IC50 = 22 nM T79031 CGO28J 68321924 EC50 = 94 nM T79031 C84FKJ 68321947 EC50 = 47 nM T79031 CFTJ53 68322072 EC50 = 86 nM T79031 C0TZ4R 68322076 IC50 = 24 nM T79031 CLNG90 68322078 IC50 = 74 nM T79031 CA15JL 68322079 EC50 = 136 nM T79031 C81GAK 68322085 EC50 = 119 nM T79031 CP98HL 68322184 EC50 = 110 nM T79031 C7I8VG 68322203 IC50 = 604 nM T79031 CP8FQ7 68352447 IC50 = 19 nM T79031 CR8TC4 68353987 IC50 = 27 nM T79031 C56CFA 68448803 IC50 > 10000 nM T79031 CPO3Q9 68691806 IC50 = 4 nM T79031 CSG7D2 68693259 IC50 = 6.5 nM T79031 CKDX07 68693809 IC50 = 3.6 nM T79031 CX1W5L 68694228 IC50 > 40000 nM T79031 C59PTV 68694939 IC50 = 9.3 nM T79031 C4GU7N 68695405 IC50 = 65 nM T79031 C4MUK2 68695669 IC50 = 4 nM T79031 CL4AV7 68695878 IC50 = 3.6 nM T79031 CQG75W 68696955 IC50 = 7 nM T79031 C0SI4O 68696972 IC50 = 160 nM T79031 C53IHQ 68696989 IC50 = 92 nM T79031 CE0FJ1 68697394 IC50 = 8.3 nM T79031 CD0B4L 68697749 IC50 = 30500 nM T79031 C3A1RB 68697829 IC50 = 5 nM T79031 C7G6CR 68698423 IC50 = 2.4 nM T79031 C70QEL 68698631 IC50 = 11 nM T79031 CL9T6R 68699050 IC50 = 2.2 nM T79031 C60VEF 68699589 IC50 = 29 nM T79031 CP5CH8 68700798 IC50 = 2 nM T79031 CDQE76 70132509 Ki = 3821 nM T79031 C3CSE7 70169280 IC50 = 73 nM T79031 CI8W6M 70356221 IC50 = 77 nM T79031 C6LA2T 70356350 IC50 = 2 nM T79031 C9KBS1 70374550 IC50 = 12 nM T79031 CC4V3Z 70374972 IC50 = 3 nM T79031 CTO36I 70680446 IC50 = 80 nM T79031 CDX40V 70680447 IC50 = 100 nM T79031 C9F1QE 70680448 IC50 = 73 nM T79031 CR8E1S 70681035 Ki = 550 nM T79031 CK12BH 70681036 Ki = 80 nM T79031 CX3F1O 70681037 Ki = 1700 nM T79031 CCZ5J0 70681598 IC50 = 8 nM T79031 COE50A 70681599 IC50 = 4 nM T79031 C9IBN5 70681952 IC50 = 8900 nM T79031 C23QAJ 70682005 IC50 = 34 nM T79031 C3BZY2 70682174 IC50 = 36100 nM T79031 CG4DK9 70682176 IC50 = 6660 nM T79031 C4L3CR 70682280 Ki = 104 nM T79031 C52DZA 70683157 Ki = 720 nM T79031 C3TO8Q 70684053 IC50 = 7.7 nM T79031 C1MJX6 70684054 IC50 = 0.15 nM T79031 CI03XR 70684068 IC50 = 11100 nM T79031 C68JCR 70684121 IC50 = 25 nM T79031 CV84NM 70684257 IC50 = 6740 nM T79031 CF2K3Y 70684265 IC50 > 30000 nM T79031 C3JT2H 70684273 IC50 = 10500 nM T79031 C6S9KL 70684278 IC50 = 21400 nM T79031 CATH92 70684290 IC50 = 9600 nM T79031 C3QB0U 70684356 Ki = 13 nM T79031 C7E3KO 70685235 Ki = 370 nM T79031 C4HWC5 70685236 Ki = 110 nM T79031 C9JS8A 70686192 IC50 = 270 nM T79031 C4H3IE 70686193 IC50 = 220 nM T79031 CZ5UA1 70686194 IC50 = 2300 nM T79031 CL1EZ3 70686213 IC50 = 600 nM T79031 CJ4ZN8 70686411 IC50 = 7380 nM T79031 C4CI1N 70686435 IC50 = 15200 nM T79031 C9APE1 70686436 IC50 = 5360 nM T79031 C7HU4P 70686438 IC50 = 13600 nM T79031 CH35YM 70687977 IC50 = 6.6 nM T79031 CHD86L 70687986 IC50 = 2 nM T79031 C2T5EQ 70688326 IC50 = 180 nM T79031 C73WJM 70688498 IC50 = 4000 nM T79031 CIA5Q8 70688505 IC50 = 7520 nM T79031 C8WBS4 70688511 IC50 = 8820 nM T79031 CEI5D1 70688538 IC50 = 25400 nM T79031 C5EQN6 70688624 Ki = 122 nM T79031 CQTH20 70688625 Ki = 11 nM T79031 C26VKR 70688626 Ki = 39 nM T79031 CV1DC5 70689418 IC50 = 4900 nM T79031 CMQ0T5 70690011 IC50 = 0.7 nM T79031 CN8ZQ9 70690351 IC50 = 1700 nM T79031 C0F1WT 70690399 IC50 = 192 nM T79031 C97SAZ 70690400 IC50 = 67 nM T79031 CD90RL 70690401 IC50 = 13 nM T79031 C3KTC7 70690563 IC50 = 7980 nM T79031 C2JPZ3 70690564 IC50 > 50000 nM T79031 CQW43C 70690565 IC50 = 4310 nM T79031 CUJT39 70690591 IC50 = 11000 nM T79031 C7CJ9K 70690592 IC50 = 8280 nM T79031 CX49OI 70690595 IC50 = 10300 nM T79031 CR2KV1 70690689 Ki = 106 nM T79031 CR57LJ 70692159 IC50 = 6 nM T79031 CU56RG 70692503 IC50 = 5300 nM T79031 CW28IQ 70692504 IC50 = 16 nM T79031 CW3C7D 70692572 IC50 = 122 nM T79031 CO2YW8 70692714 IC50 > 100000 nM T79031 C8I1QH 70692833 Ki = 79 nM T79031 CL97IX 70692834 Ki = 144 nM T79031 CHD69G 70693646 Ki = 6000 nM T79031 CKBI78 70694545 IC50 = 2.3 nM T79031 CIS6W4 70694546 IC50 = 4.6 nM T79031 CM7RF4 70694547 IC50 = 6.9 nM T79031 CXN0B2 70694548 IC50 > 10000 nM T79031 C1CLT7 70694566 IC50 = 3200 nM T79031 CVG1W5 70694577 IC50 = 1400 nM T79031 CKRV32 70694755 IC50 = 15700 nM T79031 CFU45O 70694765 IC50 = 7520 nM T79031 C8VRP5 70694784 IC50 = 10700 nM T79031 CIG9N7 70694863 Ki = 23 nM T79031 CL4HT8 70695762 Ki = 310 nM T79031 CT25CI 70696325 IC50 = 8 nM T79031 CY03PS 70696614 IC50 = 600 nM T79031 CEB7M8 70696663 IC50 = 19 nM T79031 CNF49O 70696795 IC50 = 13600 nM T79031 CLA17Z 70696796 IC50 = 45600 nM T79031 C1H5VR 70696798 IC50 = 5390 nM T79031 CWD1B4 70696799 IC50 > 80000 nM T79031 C7JLX6 70696804 IC50 = 10100 nM T79031 CLY3B9 70696917 Ki = 163.8 nM T79031 CQ4LR7 71112644 IC50 = 49 nM T79031 C9E7QP 71112763 IC50 = 9 nM T79031 CJ0H3F 71183876 IC50 = 31 nM T79031 CAUH23 71183901 IC50 = 50 nM T79031 CBV36S 71183925 IC50 = 60 nM T79031 C1ZW9L 71183951 IC50 = 2 nM T79031 C7O5IT 71268741 IC50 = 61 nM T79031 CZ9LT5 71268850 IC50 = 5100 nM T79031 CG5MW2 71273898 IC50 = 18 nM T79031 CE69IS 71273947 IC50 = 100 nM T79031 CQD14Z 71274016 IC50 = 29 nM T79031 CY5NV8 71274019 IC50 = 12 nM T79031 CES40A 71305034 IC50 = 184 nM T79031 CLDW48 71305057 IC50 = 19 nM T79031 C13JDK 71305059 IC50 = 776 nM T79031 CB85AL 71305060 IC50 = 40 nM T79031 CE48HC 71305061 IC50 = 10 nM T79031 CTD7W8 71310633 IC50 = 136150 nM T79031 C54CLM 71449357 Ki = 8 nM T79031 C7LWE4 71449474 IC50 = 46.77 nM T79031 COT91L 71449475 IC50 = 8 nM T79031 CS6V0J 71449476 IC50 = 4 nM T79031 CEV0B7 71449561 IC50 = 8.5 nM T79031 CV3IR8 71449803 IC50 = 1114000 nM T79031 C92TEK 71449804 IC50 = 1848000 nM T79031 CX2TS0 71449805 IC50 > 200000 nM T79031 C92RIS 71449970 IC50 = 0.76 nM T79031 CHU5V7 71449971 IC50 = 0.15 nM T79031 CL64JH 71449972 IC50 = 2.1 nM T79031 C21OKC 71449973 IC50 = 900 nM T79031 CUIL24 71449974 IC50 = 2820 nM T79031 C4W8ER 71450028 Ki = 9 nM T79031 CS28FT 71450031 Ki = 10 nM T79031 C3SN9M 71450032 Ki = 4 nM T79031 CU8S0P 71450033 Ki > 10000 nM T79031 C93KRD 71450105 Ki = 7.2 nM T79031 C1C6UV 71450309 IC50 = 15 nM T79031 CR9W1Q 71450310 IC50 = 11 nM T79031 C08RHF 71450318 IC50 = 14000 nM T79031 CMK0J1 71450319 IC50 = 29500 nM T79031 CP9WH2 71451161 Ki = 33 nM T79031 C5SJ7V 71451280 IC50 = 44.67 nM T79031 C86RHK 71451365 IC50 > 10000 nM T79031 CVKC68 71451473 IC50 = 310 nM T79031 CP9L3W 71451612 IC50 = 50700 nM T79031 CVR4A2 71451687 IC50 = 28 nM T79031 C8MT7W 71451786 IC50 = 116000 nM T79031 CSD40U 71451787 IC50 = 34100 nM T79031 C7V3QB 71451788 IC50 = 24300 nM T79031 CIF8L6 71451795 IC50 = 1210 nM T79031 C2O0LB 71451796 IC50 = 5280 nM T79031 CL7P2A 71451832 IC50 = 8.64 nM T79031 C7MAL1 71451851 IC50 = 10 nM T79031 C2AB9Q 71451852 Ki = 30 nM T79031 C5VDH0 71451853 Ki = 30 nM T79031 CV6C5O 71451854 Ki = 2400 nM T79031 C2IL4C 71451855 Ki > 10000 nM T79031 C49JDX 71451915 Ki = 7.3 nM T79031 CDQ09Y 71452058 IC50 > 10000 nM T79031 CN26XZ 71452059 IC50 > 10000 nM T79031 CA3H9D 71452060 IC50 > 10000 nM T79031 C2UC7A 71452061 IC50 = 124 nM T79031 C49HNE 71452117 IC50 = 69.5 nM T79031 CFZU38 71452124 IC50 = 12 nM T79031 CJD48Q 71452125 IC50 = 11 nM T79031 CJ8IK3 71452990 IC50 = 370 nM T79031 C83YMC 71452994 IC50 = 4.5 nM T79031 C9J4FO 71453097 IC50 = 7.8 nM T79031 C5CK7V 71453297 IC50 = 85000 nM T79031 CXT9Y4 71453445 IC50 = 59900 nM T79031 C8Z7NF 71453446 IC50 = 39400 nM T79031 CL5RC7 71453447 IC50 = 14100 nM T79031 C09HJT 71453520 IC50 = 30 nM T79031 CPDE37 71453601 IC50 = 12600 nM T79031 C90LIQ 71453602 IC50 = 14300 nM T79031 C71TCV 71453603 IC50 = 23200 nM T79031 C45PHI 71453617 IC50 = 2.59 nM T79031 C3X9OY 71453618 IC50 = 2510 nM T79031 CPOW01 71453619 IC50 = 2020 nM T79031 CEB6T9 71453620 IC50 = 280 nM T79031 CRN7T4 71453665 Ki = 2 nM T79031 CW52OF 71453667 Ki = 430 nM T79031 C8G5JE 71453668 Ki = 850 nM T79031 CLT04G 71453669 Ki = 40 nM T79031 C87MJF 71453670 Ki = 50 nM T79031 C3PNQ1 71453671 Ki = 60 nM T79031 CSK04F 71453672 Ki = 1800 nM T79031 CLM96W 71453702 Ki = 7 nM T79031 CNS4F1 71453708 Ki = 8800 nM T79031 CTV35W 71453879 IC50 > 10000 nM T79031 CLE7P2 71453880 IC50 = 54.2 nM T79031 CO67FA 71453881 IC50 = 48.8 nM T79031 CXEQ42 71453953 IC50 = 47 nM T79031 C7I0FT 71453954 IC50 = 71 nM T79031 C2K4HT 71454734 IC50 = 8.8 nM T79031 CKC09J 71454735 Ki = 47 nM T79031 CK5NM4 71454736 IC50 = 26 nM T79031 CC9Z6T 71454827 IC50 > 30199.52 nM T79031 CU59JM 71454828 IC50 = 4 nM T79031 CJX7L1 71454829 IC50 = 3083.85 nM T79031 CF9N6A 71455157 IC50 = 165000 nM T79031 CMKO02 71455334 IC50 = 20600 nM T79031 CFQ4O6 71455339 IC50 = 7000 nM T79031 C4IOH6 71455340 IC50 = 2240 nM T79031 C8J1LO 71455341 IC50 = 2110 nM T79031 CH46YF 71455353 IC50 = 2200 nM T79031 C23UVY 71455394 Ki = 132 nM T79031 CY8N9H 71455395 Ki = 280 nM T79031 CLDM01 71455396 Ki = 10 nM T79031 C4D8HF 71455397 Ki = 30 nM T79031 CR9VU6 71455427 Ki = 6 nM T79031 C2NM4Q 71455471 IC50 = 9.5 nM T79031 C93BQC 71455611 IC50 = 5430 nM T79031 CREI47 71455687 IC50 = 22.8 nM T79031 CJGT17 71455688 IC50 = 5.4 nM T79031 CCM0I6 71455697 IC50 = 6000 nM T79031 C05OTM 71455788 IC50 = 1.6 nM T79031 C3D6BK 71456273 IC50 = 1058 nM T79031 CIY08V 71456491 Ki = 9500 nM T79031 CGB0O1 71456492 Ki = 44000 nM T79031 CYGD69 71456609 IC50 = 38.9 nM T79031 CC7F6N 71456803 IC50 > 100000 nM T79031 C2B8LY 71456805 IC50 > 100000 nM T79031 CWG67A 71456949 IC50 = 24500 nM T79031 CS9UN7 71456950 IC50 > 200000 nM T79031 C7RF3G 71456951 IC50 = 25600 nM T79031 C98YES 71456952 IC50 = 119000 nM T79031 CH30NP 71457108 IC50 = 11000 nM T79031 C0UVB5 71457116 IC50 = 39 nM T79031 CMB6O8 71457147 IC50 = 2.97 nM T79031 COF9B5 71457165 IC50 = 91 nM T79031 CB9PI6 71457166 Ki = 2 nM T79031 C78UTY 71457167 Ki = 15 nM T79031 CUDF46 71457168 Ki = 10 nM T79031 CK28SL 71457169 Ki = 280 nM T79031 CUG45M 71457170 Ki = 50 nM T79031 C0ZT7J 71457171 Ki = 20 nM T79031 CZ80AH 71457172 Ki = 6 nM T79031 C7KP0W 71457173 Ki = 1700 nM T79031 C36TJY 71457202 Ki = 64 nM T79031 C4O2GZ 71457203 Ki = 4 nM T79031 CWA79L 71457260 Ki = 0.4 nM T79031 CL2S3Y 71457261 Ki = 0.47 nM T79031 CK73LU 71457396 IC50 = 211 nM T79031 C3LFE2 71457462 IC50 = 812 nM T79031 CO3ID7 71457465 IC50 = 35.2 nM T79031 CH6Q3P 71457466 IC50 = 5.7 nM T79031 CCFZ37 71457467 IC50 = 3.4 nM T79031 CS18XN 71457468 IC50 = 3.2 nM T79031 CC9T2S 71458462 IC50 = 8.9 nM T79031 CNM98L 71458534 IC50 = 99 nM T79031 CS48ZA 71458535 IC50 = 290 nM T79031 CS1WK4 71458818 IC50 = 502000 nM T79031 CY59BM 71458819 IC50 = 103000 nM T79031 CJTC95 71458820 IC50 = 46500 nM T79031 C03WEO 71458974 IC50 = 14000 nM T79031 CQ1G2L 71458975 IC50 = 14900 nM T79031 C7V4WH 71458976 IC50 = 9100 nM T79031 CM80QT 71458988 IC50 = 2520 nM T79031 CY50WM 71459034 Ki = 1 nM T79031 CM86PY 71459036 Ki = 1800 nM T79031 C9GX1E 71459037 Ki > 5000 nM T79031 CG1NF5 71459038 Ki = 910 nM T79031 CLG93R 71459108 Ki = 0.036 nM T79031 CJ98EQ 71459165 IC50 = 32000 nM T79031 CYL5C6 71459166 IC50 = 18000 nM T79031 C58BIQ 71459167 IC50 = 2100 nM T79031 CV4ZI2 71459168 IC50 = 14 nM T79031 C0BA3U 71459341 IC50 = 76.6 nM T79031 CN8I4U 71459342 IC50 = 5.5 nM T79031 CDKZ36 71459343 IC50 = 3.7 nM T79031 C0HD3K 71459395 IC50 = 27 nM T79031 CQC6U3 71460181 Ki = 22000 nM T79031 CH3G9B 71460182 IC50 = 81 nM T79031 C3MV5B 71460183 IC50 = 3.1 nM T79031 CV0E9B 71460380 IC50 = 12 nM T79031 CBO2M4 71460381 IC50 = 230 nM T79031 C6OC0Z 71460382 IC50 = 44 nM T79031 CPC9D4 71460630 IC50 = 619000 nM T79031 CMF68W 71460696 IC50 = 69 nM T79031 CXC75B 71460773 IC50 = 10200 nM T79031 CET27N 71460783 IC50 = 1880 nM T79031 C8RLW4 71460789 IC50 = 770 nM T79031 CE1U2X 71460835 Ki = 1200 nM T79031 C85AJU 71460836 Ki = 140 nM T79031 CK18LM 71460837 Ki = 50 nM T79031 C0NJ6Y 71460877 Ki = 11 nM T79031 CFQ16C 71460916 Ki > 1000 nM T79031 C1PRD6 71461037 IC50 > 10000 nM T79031 C9L1IU 71461038 IC50 = 166 nM T79031 CH72YK 71461109 IC50 = 5.2 nM T79031 CBMS65 71461110 IC50 = 29 nM T79031 CC94IF 71461117 IC50 = 1000 nM T79031 CP6IV2 71462074 IC50 = 19 nM T79031 CD4QU0 71462075 IC50 = 5600 nM T79031 C5IQM8 71462336 IC50 = 70000 nM T79031 CI5C1R 71462337 IC50 > 2000000 nM T79031 CH78MO 71462338 IC50 = 614000 nM T79031 CP7E9G 71462339 IC50 = 59000 nM T79031 CJQ85O 71462340 IC50 = 53300 nM T79031 CN6M7B 71462407 IC50 = 33 nM T79031 C1NJP6 71462501 IC50 = 54000 nM T79031 C50VTC 71462510 IC50 = 1780 nM T79031 CL21DT 71462547 Ki = 8 nM T79031 C21LOE 71462548 Ki = 20 nM T79031 C4NR7K 71462580 Ki = 4000 nM T79031 CMHS87 71462611 Ki = 25 nM T79031 CP18GA 71462843 IC50 = 26.1 nM T79031 C8F6LX 71462849 IC50 = 64.3 nM T79031 C2Q4VT 71462850 IC50 = 9.5 nM T79031 CUD3K5 71462851 IC50 = 2.9 nM T79031 CG9N3H 71462852 IC50 = 16 nM T79031 C0GBL7 71466345 IC50 = 59 nM T79031 C74VXH 71466346 IC50 = 15 nM T79031 C5JR4E 71466347 IC50 = 7.9 nM T79031 C2Z6UE 71468021 Ki = 27.2 nM T79031 C1T8BI 71479644 IC50 = 20 nM T79031 CD95AJ 71486743 IC50 = 12 nM T79031 CC3N4O 71492530 Ki = 1 nM T79031 CK20MH 71502737 IC50 = 31 nM T79031 CD70GQ 71516860 IC50 = 1.7 nM T79031 CFG2R8 71518025 IC50 = 35000 nM T79031 C78SCW 71518195 IC50 = 10900 nM T79031 C3C1TY 71518196 IC50 = 12500 nM T79031 C4WC0M 71518361 IC50 = 4900 nM T79031 CNSP16 71518362 IC50 = 2400 nM T79031 C6V0DB 71518363 IC50 > 1200 nM T79031 C6YTR8 71518684 IC50 = 43000 nM T79031 C6ITD8 71518685 IC50 = 2600 nM T79031 C60OUP 71518848 IC50 = 4200 nM T79031 C1FL6A 71529262 IC50 = 35 nM T79031 C10UQB 71529265 IC50 = 830 nM T79031 CB8DU6 71529426 IC50 = 19 nM T79031 CBO09H 71529465 IC50 = 12 nM T79031 CV9X7J 71532069 IC50 = 8.4 nM T79031 C18EPN 71548079 IC50 = 0.031 nM T79031 C9A1FX 71550071 IC50 = 1.1 nM T79031 CD6QA1 71550203 IC50 = 168 nM T79031 CRG0L2 71571523 IC50 = 96 nM T79031 CY36RO 71572417 IC50 = 22200 nM T79031 C3RS8D 71581444 IC50 = 17 nM T79031 CJ9S3O 71581445 IC50 = 54 nM T79031 C5N8FV 71582886 IC50 = 119 nM T79031 CIKQ69 71582887 IC50 = 578 nM T79031 CTVI47 71582888 IC50 = 98 nM T79031 CMA86X 71582889 IC50 = 326 nM T79031 CU8QX2 71582923 IC50 = 101000 nM T79031 CLS5E7 71582924 IC50 = 58900 nM T79031 C8BT4H 71582925 IC50 > 100000 nM T79031 COF5Y0 71582986 IC50 = 854 nM T79031 CCAN72 71582987 IC50 = 928 nM T79031 C4MYB7 71582988 IC50 > 10000 nM T79031 CYD78S 71582989 IC50 > 10000 nM T79031 CNDT59 71583021 IC50 > 100000 nM T79031 CUB68J 71583022 IC50 = 63300 nM T79031 CB3A6O 71583023 IC50 > 100000 nM T79031 C0G2RX 71583025 IC50 > 100000 nM T79031 CW9JL2 71583097 IC50 = 25740 nM T79031 C2E1MI 71583098 IC50 = 26430 nM T79031 C8Z9DI 71583099 IC50 = 741 nM T79031 C3M8CI 71583100 IC50 = 3550 nM T79031 CP7CV0 71584475 IC50 = 9267 nM T79031 C74SQB 71584476 IC50 = 1216 nM T79031 CEU83G 71584477 IC50 > 10000 nM T79031 C0V6NI 71584478 IC50 > 10000 nM T79031 C0B1QM 71584523 IC50 = 323000 nM T79031 CB2UL3 71584525 IC50 > 100000 nM T79031 CYSA30 71584604 IC50 = 503 nM T79031 C52ERF 71584605 IC50 = 9810 nM T79031 CGQ96N 71584606 IC50 > 10000 nM T79031 CB32QX 71584607 IC50 = 849 nM T79031 CAR43K 71584608 IC50 > 10000 nM T79031 CS0Y6K 71584645 IC50 > 100000 nM T79031 C1NP5F 71584646 IC50 = 77100 nM T79031 CXO41P 71584647 IC50 = 85700 nM T79031 C63BJM 71584648 IC50 = 33500 nM T79031 C6S0IQ 71584649 IC50 = 26900 nM T79031 CGET05 71584650 IC50 = 63900 nM T79031 C89CZA 71598542 IC50 = 36 nM T79031 C6N4LP 71598543 IC50 = 210 nM T79031 CT68JM 71614688 IC50 = 39400 nM T79031 C2IE6X 71614689 IC50 = 74900 nM T79031 C8H4SR 71614690 IC50 = 47500 nM T79031 CKOA54 71614691 IC50 > 200000 nM T79031 CE06BZ 71614885 IC50 > 200000 nM T79031 C0GU7X 71614886 IC50 = 72400 nM T79031 CMKO95 71614887 IC50 = 30800 nM T79031 CPAK75 71614888 IC50 = 84900 nM T79031 CKY13T 71614889 IC50 > 200000 nM T79031 C3J1DC 71614890 IC50 > 200000 nM T79031 CAB52T 71614891 IC50 > 200000 nM T79031 C9MO3W 71615087 IC50 > 200000 nM T79031 C49BJF 71615088 IC50 = 120000 nM T79031 CWC86H 71615089 IC50 > 200000 nM T79031 CUT7V2 71615090 IC50 > 200000 nM T79031 CVU74Y 71615091 IC50 = 100000 nM T79031 C0PEJ5 71615092 IC50 > 200000 nM T79031 CIGV69 71619629 IC50 = 1 nM T79031 CHK9Y2 71624098 EC50 = 184 nM T79031 CO3YI9 71624343 IC50 = 431 nM T79031 CI97AH 71624344 IC50 = 8661 nM T79031 CYQI35 71624345 IC50 = 2363 nM T79031 CIC4L2 71624469 IC50 = 6270 nM T79031 CA9Y2O 71624470 EC50 = 30 nM T79031 CIU5Q1 71624579 IC50 = 501 nM T79031 C7Z3GY 71624580 EC50 = 188 nM T79031 C2MSD3 71624581 EC50 = 66 nM T79031 C4NHO5 71624685 IC50 = 47 nM T79031 CI6N2U 71624686 EC50 = 25 nM T79031 C5A6UZ 71624687 EC50 = 96 nM T79031 CMN85D 71624688 EC50 = 1596 nM T79031 CI5P2V 71624689 IC50 = 123 nM T79031 C6K3CN 71625880 IC50 = 68 nM T79031 CV7G9C 71663691 IC50 = 87 nM T79031 CX73JM 71663692 IC50 = 24 nM T79031 CQ57VI 71663693 IC50 = 61 nM T79031 CE4DJ8 71663694 IC50 = 54 nM T79031 C9UN3Q 71663695 IC50 = 22 nM T79031 C1H2BL 71663858 IC50 = 25 nM T79031 CCUI41 71664591 IC50 = 2 nM T79031 CKX64V 71664592 IC50 = 88 nM T79031 CGD2R7 71680685 IC50 = 400 nM T79031 CT5L2D 71680688 IC50 = 32 nM T79031 C6EDG5 71680844 IC50 = 320 nM T79031 C4CR7D 71680846 IC50 = 500 nM T79031 C4C9OW 71680849 IC50 = 7900 nM T79031 C26UGV 71681009 IC50 = 400 nM T79031 CG2F5B 71681010 IC50 = 500 nM T79031 CN7ZH6 71681015 IC50 = 20000 nM T79031 C50DHN 71681166 IC50 = 2000 nM T79031 C10OCG 71681315 IC50 = 16000 nM T79031 CRQ1Y6 71681316 IC50 = 500 nM T79031 C4OU0Y 71681318 IC50 = 320 nM T79031 C13RPX 71681468 IC50 = 5000 nM T79031 CB6TI0 71681469 IC50 = 32000 nM T79031 C16LCK 71681471 IC50 = 10000 nM T79031 C86XQA 71681473 IC50 = 790 nM T79031 CU23DO 71681634 IC50 = 40 nM T79031 C8H2PC 71681635 IC50 = 630 nM T79031 C9B2RV 71681636 IC50 = 630 nM T79031 CH4R7G 71682752 IC50 = 3200 nM T79031 CBVC07 71682893 IC50 = 320 nM T79031 CFE3Y7 71683044 IC50 = 200 nM T79031 C3ISR6 71683048 IC50 = 2000 nM T79031 CFKH23 71713792 IC50 = 200 nM T79031 C58FAK 71713793 IC50 = 1720 nM T79031 CH8P2L 71713948 IC50 = 1020 nM T79031 CVW9I8 71713949 IC50 = 210 nM T79031 CC3PG2 71713950 IC50 = 1300 nM T79031 CFY5U2 71713951 IC50 = 4000 nM T79031 CG5O9D 71713952 IC50 = 12 nM T79031 CN86TL 71713954 IC50 = 15 nM T79031 CS5BC8 71714101 IC50 = 11 nM T79031 C54DZH 71714118 IC50 = 2250 nM T79031 CP56WO 71718352 IC50 = 1 nM T79031 C6LIH9 71719178 IC50 > 11000 nM T79031 C24EOD 71719654 IC50 > 160000 nM T79031 COJ3I6 71720622 IC50 = 52 nM T79031 CPI2B3 71726571 IC50 = 45 nM T79031 C8J4WK 71726572 IC50 = 120 nM T79031 C08CYJ 71726699 IC50 = 5.9 nM T79031 C38LNQ 71726700 IC50 = 5.9 nM T79031 CPX7C6 71726820 IC50 = 2.7 nM T79031 CN2V1S 71738909 Ki > 10000 nM T79031 COVS02 71812189 IC50 = 3 nM T79031 CLE0M5 71814501 IC50 = 148 nM T79031 CF9Q6G 71814502 IC50 = 186 nM T79031 C8GBJ2 71814503 IC50 = 60 nM T79031 C8OAN7 71814504 IC50 = 1300 nM T79031 CVFW51 71814680 IC50 = 221 nM T79031 C53EOF 71814681 IC50 = 1325 nM T79031 C1W4ND 71814682 IC50 = 858 nM T79031 CTG12Z 71814683 IC50 = 8 nM T79031 C5NXB9 71815029 IC50 = 9 nM T79031 CGBA97 71815030 IC50 = 6 nM T79031 C1GFK3 71815031 IC50 = 89 nM T79031 C4DNQ3 71815032 IC50 = 690 nM T79031 C9UV7C 72190738 IC50 = 530 nM T79031 CZ60LS 72191037 IC50 = 33 nM T79031 C14GNR 72191038 IC50 = 8 nM T79031 C4V7UP 72191342 IC50 > 10000 nM T79031 C20HKS 72191344 IC50 = 18 nM T79031 C0C5QH 72191659 IC50 = 16 nM T79031 CYEI57 72191660 IC50 = 12 nM T79031 C36QKA 72191661 IC50 = 13 nM T79031 C1Y8VS 72191976 IC50 = 75 nM T79031 CO28LK 72191977 IC50 = 382 nM T79031 C5ZGJ6 72191978 IC50 = 226 nM T79031 C7K9YS 72204170 IC50 = 16600 nM T79031 CF9O1X 72204363 IC50 = 18000 nM T79031 CD0BU3 72204552 IC50 > 200000 nM T79031 CJ10ZV 72204554 IC50 > 200000 nM T79031 CN63JA 72204556 IC50 > 200000 nM T79031 C4U9KG 72204558 IC50 = 9300 nM T79031 CI7MT1 72204757 IC50 = 7500 nM T79031 CAT8Q9 72204758 IC50 = 3300 nM T79031 C5ZQA3 72204759 IC50 = 23300 nM T79031 C1FKW7 72204760 IC50 = 8400 nM T79031 C1JB3V 72204761 IC50 = 20800 nM T79031 C3ZL7J 72204935 IC50 = 6100 nM T79031 CIXD45 72204936 IC50 = 7500 nM T79031 CC8D4V 72204937 IC50 = 11800 nM T79031 C8O3ID 72204938 IC50 = 4000 nM T79031 CCJ2L5 72204939 IC50 = 2900 nM T79031 CO5MH1 72204940 IC50 > 200000 nM T79031 CGJ7X2 72205116 IC50 = 132000 nM T79031 CS7TH5 72205117 IC50 > 200000 nM T79031 CU80HY 72547065 IC50 = 614 nM T79031 CE3X8Y 72547066 IC50 = 4 nM T79031 CCVG84 72547070 IC50 = 6 nM T79031 CX70JT 72547320 IC50 = 4 nM T79031 C7S2TU 72696067 IC50 = 4660 nM T79031 C8ZCE4 72697998 IC50 = 6780 nM T79031 CI1GL7 72698000 IC50 = 4210 nM T79031 CAP0H5 72698148 IC50 = 4270 nM T79031 C0KYO6 72943702 IC50 = 2.2 nM T79031 C5DC0Z 72946535 IC50 = 660 nM T79031 C09DKS 72946536 IC50 = 720 nM T79031 C8K6NI 72946537 IC50 = 390 nM T79031 CZ0W2F 72946538 IC50 = 570 nM T79031 CD7Y8W 72946737 IC50 = 450 nM T79031 CQM8U4 72946738 IC50 = 50 nM T79031 CTH7B3 72946739 IC50 = 440 nM T79031 CZ9FI5 72946741 IC50 = 360 nM T79031 CQ3DV8 72946943 IC50 = 70 nM T79031 C6TR1J 72946944 IC50 = 1350 nM T79031 CX40JE 72946945 IC50 = 670 nM T79031 C82DSO 72946946 IC50 = 720 nM T79031 CNL10Y 72947155 IC50 = 3150 nM T79031 CYXC78 72947373 IC50 = 120 nM T79031 C4HIV9 72947374 IC50 = 730 nM T79031 CEA3N2 72947375 IC50 > 5000 nM T79031 CJW1K5 72947376 IC50 = 640 nM T79031 C8FKH3 72947377 IC50 = 480 nM T79031 C2TZY0 72947378 IC50 > 5000 nM T79031 CL8ZX4 72947563 IC50 > 5000 nM T79031 CXB6V2 73212455 IC50 = 151 nM T79031 CA1GF7 73212458 IC50 = 89 nM T79031 C98ONY 73212532 IC50 = 79 nM T79031 C48RAF 73213042 IC50 = 1800000 nM T79031 C52QYP 73213044 IC50 = 1400000 nM T79031 C8DSX2 73213045 IC50 = 250000 nM T79031 C3W0YC 73213128 IC50 = 450000 nM T79031 C6DF7G 73345437 IC50 = 60000 nM T79031 C43EOP 73345995 IC50 = 4.7 nM T79031 CEHO98 73345996 IC50 = 120 nM T79031 CMHA87 73346002 IC50 = 2 nM T79031 C1IFV6 73346019 IC50 = 42 nM T79031 CI3U9L 73346530 IC50 > 200000 nM T79031 C62BWK 73347547 IC50 = 6 nM T79031 C7W5ER 73348463 IC50 > 200000 nM T79031 CU7W6R 73348464 IC50 = 20000 nM T79031 C35IFQ 73349076 IC50 = 19700 nM T79031 CK40LM 73349243 IC50 = 7 nM T79031 COT85D 73350046 IC50 = 2000 nM T79031 CDK36B 73350049 IC50 = 2500 nM T79031 CR2JN8 73350632 IC50 = 110 nM T79031 C3ABQ1 73350653 IC50 = 116 nM T79031 CSWI58 73350654 IC50 = 15 nM T79031 C2PLM7 73350655 IC50 = 574 nM T79031 C6LS2M 73351114 IC50 = 41400 nM T79031 C76QTO 73351551 IC50 = 9000 nM T79031 CWE51A 73352121 IC50 = 25 nM T79031 CSM21F 73352126 IC50 = 81 nM T79031 CDQ52R 73352584 IC50 > 200000 nM T79031 CE7U0M 73353004 IC50 = 1200 nM T79031 CMB8W4 73353577 IC50 = 140 nM T79031 C5RL3S 73353578 IC50 = 67 nM T79031 CG0YR8 73354162 IC50 = 3 nM T79031 CQHV29 73354525 IC50 > 100000 nM T79031 C1GUY0 73354529 IC50 = 40 nM T79031 C6Z4MB 73354727 Ki = 0.3 nM T79031 C8MEY2 73355084 IC50 = 37 nM T79031 CF0ST3 73355087 IC50 = 10 nM T79031 C74BWF 73355106 IC50 = 9 nM T79031 CVW0J5 73355107 IC50 = 22 nM T79031 C27PAD 73355601 IC50 = 1300 nM T79031 CY71ES 73356167 IC50 = 30 nM T79031 C86UGE 73356659 IC50 = 5.1 nM T79031 C6VCF3 73356671 IC50 = 27105 nM T79031 C3BF0T 73356672 IC50 = 4705 nM T79031 CX7P2O 73356673 IC50 = 378 nM T79031 C0LF9I 73356861 IC50 = 150000 nM T79031 CZ6Q1I 73388368 IC50 = 25 nM T79031 CB7J0I 73507165 IC50 = 670 nM T79031 CEP9F4 73507167 IC50 = 39 nM T79031 C38SOV 73507168 IC50 = 800 nM T79031 C7Y5QC 73507384 IC50 = 30 nM T79031 CI58HT 74222429 IC50 = 0.58 nM T79031 C1X0ME 75593273 IC50 = 300 nM T79031 C97WEM 75593288 IC50 > 100000 nM T79031 CLYH10 75593331 Ki = 1 nM T79031 CD4IX1 75593344 IC50 = 24 nM T79031 CLM3N4 76309803 IC50 = 18100 nM T79031 CT8R2Z 76311036 IC50 = 5.1 nM T79031 CTG78Z 76311037 IC50 = 79 nM T79031 CWFI38 76313404 Ki = 7998.34 nM T79031 C1P7SH 76313523 IC50 = 4900 nM T79031 C16WUE 76314667 IC50 = 1.6 nM T79031 CLFK92 76316916 Ki = 3133285.72 nM T79031 C2F0ZL 76316917 Ki = 50118.72 nM T79031 CS92HG 76317036 IC50 = 7500 nM T79031 C51UAX 76318242 IC50 = 11 nM T79031 CWB7S5 76320641 Ki = 22438819.24 nM T79031 C6R0EF 76320744 IC50 = 9200 nM T79031 CA6FV4 76320745 IC50 = 6400 nM T79031 C4MF7L 76321932 IC50 = 29 nM T79031 CR4A3H 76324291 Ki = 9397.23 nM T79031 C9GW8A 76327856 Ki = 61376.2 nM T79031 C2N1OW 76327857 Ki = 5807644.18 nM T79031 C01UQY 76327955 IC50 = 14800 nM T79031 C31GTN 76329120 IC50 = 33 nM T79031 C9DLB2 76331514 Ki = 10495424.29 nM T79031 CG2V8C 76331607 IC50 = 12800 nM T79031 CR97QB 76331609 IC50 = 14300 nM T79031 COFK24 76332783 IC50 = 330 nM T79031 C2YJ4G 76335122 Ki = 1129795.91 nM T79031 CBH89U 76335123 Ki = 5902.01 nM T79031 CKX31E 76335235 IC50 = 14900 nM T79031 CUF56O 76335236 IC50 = 4700 nM T79031 C3SQ0F 76335237 IC50 = 5200 nM T79031 CTJG92 76336403 IC50 = 99 nM T79031 CQT14W 76955651 IC50 = 15 nM T79031 CJ29RM 77461103 IC50 = 3.4 nM T79031 CD1E7Y 78210254 IC50 = 0.615 nM T79031 CAUF19 78319722 IC50 = 70 nM T79031 CKOU34 78319724 IC50 = 17 nM T79031 C86QLE 81689770 IC50 = 7.6 nM T79031 CI5GO1 83453608 IC50 = 5900 nM T79031 CEQ36D 84973151 Ki = 12.9 nM T79031 CO57IZ 84973152 Ki = 81.4 nM T79031 C0X1HW 85470889 Ki = 5 nM T79031 C8EK2Y 85471653 Ki = 6.1 nM T79031 CC2T7G 86291837 IC50 = 3.9 nM T79031 C5XON4 86293009 IC50 = 3.981 nM T79031 CZLX91 86294744 IC50 = 1 nM T79031 CH12LM 86294873 IC50 = 45 nM T79031 CB5F1W 86343364 IC50 = 74 nM T79031 CKG7N2 86343365 IC50 = 7 nM T79031 C9IVM5 86343366 IC50 = 34 nM T79031 CZ7Y0L 86658490 IC50 = 320 nM T79031 CA0FL4 86699707 IC50 = 9 nM T79031 CH65UE 86762160 IC50 = 37 nM T79031 CO2RA4 86762161 IC50 = 160 nM T79031 CTS26M 86762162 IC50 = 860 nM T79031 CXL35S 86762164 IC50 = 160 nM T79031 CR5VY9 86762166 IC50 = 510 nM T79031 C7OIC6 86762648 IC50 = 0.006 nM T79031 CX34OC 86762781 IC50 = 0.482 nM T79031 CM6CG1 86765151 IC50 = 1890 nM T79031 CVD2I6 88602735 IC50 = 11 nM T79031 C4EXW3 89512662 IC50 = 4 nM T79031 CQCJ02 89512686 IC50 = 2.4 nM T79031 C1CR9M 89512731 IC50 = 1.8 nM T79031 CM61YZ 89576898 IC50 = 33 nM T79031 CRO17A 89836343 Ki = 279.9 nM T79031 CEJA29 89974871 IC50 = 5.8 nM T79031 CNY6Q0 89974884 IC50 = 6.5 nM T79031 CI4RZ9 89974885 IC50 = 31 nM T79031 C2R7VW 89974886 IC50 = 72 nM T79031 CQ89KV 89974892 IC50 = 8.4 nM T79031 C6WPY0 89974894 IC50 = 56 nM T79031 CIL02V 89974905 IC50 = 12 nM T79031 CF90DE 89974906 IC50 = 22 nM T79031 C37YXD 89976592 IC50 = 63.9 nM T79031 C0R3BF 89976659 IC50 = 34.8 nM T79031 CAKV98 89997377 IC50 = 5.6 nM T79031 CIBY41 89997417 IC50 = 9 nM T79031 C8Z9QB 89997423 IC50 = 0.4 nM T79031 C2JF6O 89997464 IC50 = 71 nM T79031 C4PT6B 89997503 IC50 = 0.9 nM T79031 CB7L1N 89997512 IC50 = 3.3 nM T79031 CE7PH6 89997520 IC50 = 0.9 nM T79031 C52QPK 89997526 IC50 = 3 nM T79031 C90TSY 89997709 IC50 = 0.8 nM T79031 C2SJY8 89997744 IC50 = 2.2 nM T79031 C7ZY4H 89997769 IC50 = 1 nM T79031 CFYO09 89997799 IC50 = 4 nM T79031 C7Z1GY 89997802 IC50 = 9 nM T79031 C89LAZ 89997856 IC50 = 10 nM T79031 C5EQM4 89997906 IC50 = 76 nM T79031 C7M5KB 89997911 IC50 = 0.5 nM T79031 CXP2Q5 89997939 IC50 = 4 nM T79031 CX4S6M 89997948 IC50 = 7 nM T79031 COR4F3 89997978 IC50 = 17 nM T79031 CDI4P0 89997990 IC50 = 4 nM T79031 C9TG4Q 89998018 IC50 = 2.3 nM T79031 CN0DA6 89998034 IC50 = 0.8 nM T79031 CD1VM9 89998106 IC50 = 1.2 nM T79031 CT38QK 89998122 IC50 = 25.3 nM T79031 CMO1B0 89998184 IC50 = 6 nM T79031 CZ5QN1 89998216 IC50 = 248 nM T79031 C7NA0W 89998237 IC50 = 3.8 nM T79031 C17DCR 90147187 IC50 = 120 nM T79031 CG5O1Y 90238856 IC50 = 290 nM T79031 C64CQV 90253299 IC50 = 22 nM T79031 CDB0K1 90253302 IC50 = 300 nM T79031 CC9JA1 90253303 IC50 = 5 nM T79031 CXB2K9 90253304 IC50 = 60 nM T79031 CQM3K5 90253316 IC50 = 70 nM T79031 CV3I1M 90253319 IC50 = 87 nM T79031 CFD37J 90253342 IC50 = 30 nM T79031 CLNT58 90253364 IC50 = 1100 nM T79031 CD6TF7 90253366 IC50 = 8 nM T79031 C8YSR3 90253370 IC50 = 350 nM T79031 CZ6AM3 90253371 IC50 = 110 nM T79031 CRN8G1 90253396 IC50 = 310 nM T79031 CJT7E3 90253397 IC50 = 150 nM T79031 C7PO1W 90308598 IC50 = 2 nM T79031 CL5A4D 90411856 IC50 = 41000 nM T79031 C6W9CF 90411858 IC50 = 15 nM T79031 C6EQO0 90412858 IC50 = 12000 nM T79031 CN0YA2 90412860 IC50 = 59 nM T79031 C7OLJ6 90414780 IC50 = 0.6 nM T79031 CY8C1D 90644231 IC50 = 62210 nM T79031 COY0N9 90654956 IC50 = 1850 nM T79031 C03YNQ 90654957 IC50 = 7040 nM T79031 CB8S1N 90654958 IC50 = 2200 nM T79031 CMAK24 90654959 IC50 = 1610 nM T79031 CL76FO 90654960 IC50 = 7180 nM T79031 CDX3A0 90654961 IC50 = 6180 nM T79031 C9AUK3 90654962 IC50 = 11530 nM T79031 CL7PI9 90655190 IC50 = 980 nM T79031 CZ18NX 90655191 IC50 = 120 nM T79031 CH7C4F 90655192 IC50 = 80 nM T79031 CMJ31X 90655193 IC50 = 80 nM T79031 C3IZ2O 90655195 IC50 = 1190 nM T79031 CG69TU 90655196 IC50 = 1200 nM T79031 C6WH0F 90655198 IC50 = 2020 nM T79031 CPU06Y 90656183 IC50 = 0.2 nM T79031 C9Y0AL 90656184 IC50 = 20 nM T79031 C5CGK1 90656185 IC50 = 7.943 nM T79031 CMZ9C5 90656186 IC50 = 514 nM T79031 CC8B2T 90656188 IC50 = 26 nM T79031 CH0S3R 90656189 IC50 = 580 nM T79031 CB1C5A 90656190 IC50 = 1.318 nM T79031 C0V9BQ 90656191 IC50 = 36 nM T79031 CGB50T 90656192 IC50 = 20 nM T79031 C1EGV5 90656193 IC50 = 40 nM T79031 CHX6K5 90656194 IC50 = 7.2 nM T79031 C08KGC 90656195 IC50 = 25 nM T79031 CJ1R2V 90657111 IC50 = 36000 nM T79031 C1KOL2 90664301 IC50 = 1810 nM T79031 C7H6ZG 90664851 IC50 = 7300 nM T79031 CI0NQ2 90664853 IC50 = 5700 nM T79031 CLQ1F4 90664854 IC50 = 5900 nM T79031 CXB25V 90664977 IC50 = 5800 nM T79031 C1DN7L 90664978 IC50 = 6600 nM T79031 CAQ05V 90693645 Ki = 0.25 nM T79031 CCUD76 91154809 Ki = 40 nM T79031 CUI10E 91666686 IC50 = 10 nM T79031 CZJ6S7 91757962 IC50 = 599 nM T79031 CK64RW 91809482 IC50 = 72000 nM T79031 C91YPW 91809483 IC50 = 9400 nM T79031 CF3E1V 91810398 IC50 = 0.2 nM T79031 C79AZY 91824261 IC50 = 26000 nM T79031 C0ORT4 91827634 Ki = 4.3 nM T79031 CAM0G8 91864546 IC50 = 1350 nM T79031 C6CQX4 91885601 IC50 = 0.9 nM T79031 CWZX73 91971958 IC50 = 5 nM T79031 C5RF6O 101077957 IC50 > 10000 nM T79031 CSL2D7 101242500 IC50 = 2000 nM T79031 C4HLR3 101528287 IC50 > 10000 nM T79031 C6W2JF 101898808 IC50 = 17200 nM T79031 CK3V4T 109374149 IC50 > 50000 nM T79031 CSF32B 110298324 IC50 = 18.3 nM T79031 CM4DQ0 112996426 IC50 = 7900 nM T79031 CFT94I 117700435 IC50 = 11.4 nM T79031 C2P9ZX 117738849 IC50 = 6.66 nM T79031 C7Y2IL 117754251 IC50 = 10.47 nM T79031 C1UXK6 117844010 IC50 = 2 nM T79031 CLP6K8 117960375 Ki = 3 nM T79031 C6WEC5 118070156 IC50 = 1.5 nM T79031 C74EMN 118190070 Ki = 3 nM T79031 CD8NT3 118399560 IC50 = 22.8 nM T79031 C18EVY 118399566 IC50 = 27.6 nM T79031 CC7R5L 118399605 IC50 = 1.7 nM T79031 CMK5Y8 118399612 IC50 = 1.5 nM T79031 C57PSF 118399626 IC50 = 25.8 nM T79031 CN7EP4 118399635 IC50 = 27.4 nM T79031 CG4KD8 118399643 IC50 = 1.6 nM T79031 C4WAQ6 118399787 IC50 = 3.4 nM T79031 C94WRZ 118435363 IC50 = 0.64 nM T79031 C1WL4E 118435382 IC50 = 7.2 nM T79031 C5L9VH 118435403 IC50 = 3.9 nM T79031 CNXH97 118435407 IC50 = 8.2 nM T79031 C8Z2FP 118435412 IC50 = 23.7 nM T79031 CJIP45 118435414 IC50 = 12.5 nM T79031 CY6EP7 118435506 IC50 = 47.6 nM T79031 CPE35X 118435524 IC50 = 2.9 nM T79031 CVK6Y8 118435560 IC50 = 4.8 nM T79031 CN5L8K 118435601 IC50 = 0.014 nM T79031 C37SFM 118435617 IC50 = 26.9 nM T79031 C12STH 118440821 IC50 = 0.391 nM T79031 CL6IV1 118440826 IC50 = 1.9 nM T79031 CSWP40 118440832 IC50 = 0.615 nM T79031 CAXT13 118441135 IC50 = 2.1 nM T79031 C7U6ZC 118441141 IC50 = 1 nM T79031 CHIL17 118441142 IC50 = 3 nM T79031 CZLJ20 118441559 IC50 < 1 nM T79031 CR9QF7 118441560 IC50 = 13600 nM T79031 CH2JT1 118513484 IC50 = 600 nM T79031 CG7WE4 118517237 IC50 = 230 nM T79031 C98DWV 118517247 IC50 = 180 nM T79031 C19BMO 118517248 IC50 = 3700 nM T79031 CB56VQ 118577456 IC50 = 18000 nM T79031 CXZU90 118678226 IC50 = 9 nM T79031 C1J0IZ 118711805 IC50 = 40100 nM T79031 CJG10W 118711813 IC50 > 100000 nM T79031 C2Q8IE 118711815 IC50 = 22600 nM T79031 C9U5SV 118712170 IC50 = 20200 nM T79031 C9KUS7 118712171 IC50 = 42800 nM T79031 CY9G8O 118716198 IC50 > 100000 nM T79031 CL6TE3 118716321 IC50 > 100000 nM T79031 C4IZ7G 118716325 IC50 > 100000 nM T79031 CQB1N2 118716328 IC50 > 100000 nM T79031 CEU78H 118717559 IC50 > 100000 nM T79031 CCT87K 118717561 IC50 > 100000 nM T79031 CYR34C 118717562 IC50 > 100000 nM T79031 C3U5OB 118717564 IC50 > 100000 nM T79031 CSWB75 118717566 IC50 > 100000 nM T79031 C4FWD7 118717568 IC50 > 100000 nM T79031 CH87TO 118717570 IC50 > 100000 nM T79031 CXAF54 118717573 IC50 > 100000 nM T79031 CVKR02 118717582 IC50 > 100000 nM T79031 C5SZC4 118717584 IC50 > 100000 nM T79031 C50AUM 118717586 IC50 > 100000 nM T79031 CHNF21 118717648 IC50 > 100000 nM T79031 C98MHD 118717651 IC50 > 100000 nM T79031 C1UGM6 118717653 IC50 > 100000 nM T79031 CMV83O 118717655 IC50 > 100000 nM T79031 CS0T9I 118717657 IC50 > 100000 nM T79031 C1BX8S 118717659 IC50 > 100000 nM T79031 C64WVI 118717661 IC50 > 100000 nM T79031 CY96ZA 118718226 Ki = 2500.35 nM T79031 C4WHC8 118719663 Ki = 41000 nM T79031 C08UOL 118719664 Ki = 29000 nM T79031 CPT24G 118719665 Ki = 66000 nM T79031 CJW94R 118719666 Ki = 8500 nM T79031 CQ35DS 118719667 Ki = 7600 nM T79031 CP1R2J 118719668 Ki = 8500 nM T79031 CO2GZ4 118719669 Ki = 6300 nM T79031 CK1IT5 118719670 Ki = 3200 nM T79031 C5K9GN 118720051 Ki = 17000 nM T79031 CXUT34 118720052 Ki = 970 nM T79031 CRU2Q0 118720053 Ki = 12400 nM T79031 C50SLJ 118720054 Ki = 490 nM T79031 CJ19VX 118720055 Ki = 17400 nM T79031 C16QPS 118720056 Ki = 640 nM T79031 CV1Z5B 118720057 Ki = 37000 nM T79031 C0YJ7W 118720058 Ki = 22 nM T79031 CO1GD9 118720059 Ki = 14 nM T79031 CYX8Z6 118720352 IC50 = 323 nM T79031 CJKA03 118722345 IC50 = 700 nM T79031 CORN10 118722346 IC50 = 759 nM T79031 C6I4HX 118722347 IC50 = 550 nM T79031 C2GV6A 118722348 IC50 = 27 nM T79031 CRXM26 118722349 IC50 = 48 nM T79031 CVXD58 118722350 IC50 = 110 nM T79031 CJ4NR8 118722351 IC50 = 41 nM T79031 CGXN17 118722352 IC50 = 56 nM T79031 C0LUV6 118723826 IC50 = 0.7 nM T79031 CXE6I5 118723827 IC50 = 1.5 nM T79031 CKO8P6 118723828 IC50 = 2.8 nM T79031 CH95AZ 118724884 Ki = 1.6 nM T79031 C0B6US 118724885 Ki = 1640 nM T79031 CY6V9S 118724886 Ki = 471 nM T79031 CW96VR 118724887 Ki = 147.7 nM T79031 CKH83G 118724888 Ki = 201 nM T79031 C83MKX 118724889 Ki = 64.2 nM T79031 CL95VK 118724890 Ki = 192.2 nM T79031 C4PYC1 118724891 Ki = 31.9 nM T79031 C25OXU 118724892 Ki = 16.8 nM T79031 CE7ZW3 118724893 Ki = 28.9 nM T79031 C3A6VB 118725861 IC50 = 11.3 nM T79031 C3MNQ4 118725862 IC50 = 18.5 nM T79031 C1TS2W 118725863 IC50 = 1.3 nM T79031 C1LTN0 118725864 IC50 = 0.5 nM T79031 CIR0O4 118725970 IC50 = 6 nM T79031 CS6BC8 118725971 IC50 = 0.8 nM T79031 CDV7Z0 118725972 IC50 = 1.2 nM T79031 CVZ9F7 118725973 IC50 = 19 nM T79031 CX9W7R 118725974 IC50 = 0.2 nM T79031 C1X4CO 118725975 IC50 = 0.4 nM T79031 C4DVC0 118725976 IC50 = 105 nM T79031 C0SO8I 118725977 IC50 = 23 nM T79031 CN4FG2 118728007 IC50 = 870 nM T79031 C6LPG2 118728008 IC50 > 10000 nM T79031 C07WQT 118728009 IC50 = 2610 nM T79031 C9YD4G 118728010 IC50 > 10000 nM T79031 CL03SB 118728011 IC50 > 10000 nM T79031 C1ACD2 118728012 IC50 = 4460 nM T79031 CQV8E3 118728013 IC50 > 10000 nM T79031 C0QK3S 118728014 IC50 > 10000 nM T79031 CNZ5O4 118728016 IC50 > 10000 nM T79031 CWMG09 118728017 IC50 > 10000 nM T79031 C4CI1L 118728018 IC50 = 1010 nM T79031 C1COA0 118728019 IC50 > 10000 nM T79031 CSJ43T 118728020 IC50 = 480 nM T79031 CI81SM 118728021 IC50 > 10000 nM T79031 CYA1S6 118728022 IC50 > 10000 nM T79031 CUKB12 118728023 IC50 > 10000 nM T79031 CFB83M 118728024 IC50 > 10000 nM T79031 C9EP7A 118732788 IC50 = 850 nM T79031 CQD8B7 118732789 IC50 = 3940 nM T79031 C4HLF7 118732790 IC50 = 17200 nM T79031 C39IRT 118732791 IC50 = 470 nM T79031 C5VHT6 118796839 IC50 = 36 nM T79031 C64PZC 118796840 IC50 = 157 nM T79031 C4MTK9 118797904 IC50 = 9 nM T79031 C61QPW 118797905 IC50 = 0.8 nM T79031 C5W2NL 118865901 IC50 = 0.3 nM T79031 C5NE9P 118866030 IC50 = 2 nM T79031 COR8Y4 118866094 IC50 = 12 nM T79031 CELZ36 118866105 IC50 = 1.2 nM T79031 C9Z1BW 118866133 IC50 = 1.8 nM T79031 CWCX50 118866162 IC50 = 16 nM T79031 CZ7SF8 118866177 IC50 = 1.2 nM T79031 C2CZ5B 118866257 IC50 = 0.2 nM T79031 CK2U6X 118866347 IC50 = 0.4 nM T79031 CQ5Y3R 118866403 IC50 = 4.2 nM T79031 C4MLU1 118866454 IC50 = 1.3 nM T79031 CH6AT4 118866474 IC50 = 0.6 nM T79031 CA51SU 118866499 IC50 = 0.6 nM T79031 C68ELY 118866551 IC50 = 0.8 nM T79031 CGIC35 118866737 IC50 = 6.1 nM T79031 CM2N6G 118866838 IC50 = 1.1 nM T79031 CIM4Y6 118866963 IC50 = 45 nM T79031 C9M2WU 118866986 IC50 = 0.2 nM T79031 CT4Z2R 118884907 IC50 = 2.1 nM T79031 CX8JW2 118885049 IC50 = 0.7 nM T79031 CP13NA 118958876 Ki = 9.4 nM T79031 CFW1D5 118974304 Ki = 62.7 nM T79031 CRW25M 121264059 Ki = 1 nM T79031 CGH84P 121264098 Ki = 47 nM T79031 CJU2G1 121278479 IC50 = 0.6 nM T79031 C2XA0P 121298035 IC50 = 6.31 nM T79031 CO7E4P 122180108 IC50 = 1830 nM T79031 CJM51V 122180111 IC50 = 36100 nM T79031 C15DUY 122180113 IC50 = 761 nM T79031 C13ELK 122180115 IC50 = 37500 nM T79031 CXMQ41 122180117 IC50 = 21700 nM T79031 C0YHI7 122180159 IC50 = 1070 nM T79031 C5K0RY 122180160 IC50 = 230 nM T79031 C71TKE 122180161 IC50 = 980 nM T79031 C9QKP3 122180162 IC50 > 10000 nM T79031 CQL13W 122180163 IC50 > 10000 nM T79031 CMR72I 122180164 IC50 = 6910 nM T79031 CZ5VM7 122180628 Ki = 2 nM T79031 CKFA52 122180629 Ki = 1.9 nM T79031 CSN78D 122180630 Ki = 2 nM T79031 C05VYD 122180631 Ki = 1.7 nM T79031 C3BWH1 122183695 IC50 = 13400 nM T79031 CXKW60 122183696 IC50 = 11670 nM T79031 CC71VT 122183697 IC50 = 8230 nM T79031 C7K6IU 122183699 IC50 = 3210 nM T79031 CYF3K2 122183701 IC50 = 2490 nM T79031 CI1B6Q 122183702 IC50 = 5950 nM T79031 C7XMJ0 122185859 IC50 = 56000 nM T79031 CE1ZS9 122185860 IC50 = 64000 nM T79031 CMXG71 122185861 IC50 = 34000 nM T79031 CL4IP6 122185862 IC50 > 2000000 nM T79031 CB1X0A 122185863 IC50 > 1000000 nM T79031 CBE57Q 122185864 IC50 > 1000000 nM T79031 C51FVC 122185865 IC50 > 1000000 nM T79031 CZ7C2K 122185866 IC50 = 870000 nM T79031 CPUK71 122185867 IC50 > 1000000 nM T79031 C2I1FL 122185939 IC50 = 480000 nM T79031 CP0G8U 122185940 IC50 = 870000 nM T79031 C3NOH9 122185942 IC50 = 680000 nM T79031 C4K5ZM 122193027 Ki = 490 nM T79031 C15EKW 122193028 Ki = 710 nM T79031 C76XGR 122193029 Ki = 2500 nM T79031 CX7C0R 122193030 Ki = 7000 nM T79031 CEMA65 122193031 Ki = 990 nM T79031 CESW63 122193032 Ki = 2300 nM T79031 CQ9UT0 122193033 Ki = 10000 nM T79031 CG48OK 122193034 Ki = 9100 nM T79031 C8MA5T 122193035 Ki = 1400 nM T79031 C2YE4R 122193036 Ki = 150 nM T79031 C2CIN0 122193037 Ki = 450 nM T79031 CVK29T 122193038 Ki = 130 nM T79031 CC6TR4 122193039 Ki = 260 nM T79031 COK62M 122193040 Ki = 790 nM T79031 CBR63X 122193041 Ki = 610 nM T79031 CLNA26 122193042 Ki = 530 nM T79031 CI05NP 122193043 Ki = 1900 nM T79031 CC48SU 122193044 Ki = 1800 nM T79031 C4Q3WK 122193045 Ki = 420 nM T79031 CB1DI0 122193182 Ki = 560 nM T79031 C9BA5S 122193183 Ki = 230 nM T79031 C4DXM3 122193184 Ki = 220 nM T79031 C2EHL1 122193185 Ki = 20 nM T79031 CFU6Z1 122193186 Ki = 43 nM T79031 CI74XN 122193187 Ki = 25 nM T79031 CJ87GI 122193188 Ki = 3.2 nM T79031 C7PKD2 122195837 IC50 = 5.4 nM T79031 C1R4LZ 122195838 IC50 = 93 nM T79031 CSR2O7 122195839 IC50 = 9.1 nM T79031 C02BVK 122195840 IC50 = 20 nM T79031 CO3XH0 122195841 IC50 = 316 nM T79031 CKLU67 122195842 IC50 = 13 nM T79031 C28GPM 122195843 IC50 = 14 nM T79031 CW3F1J 122195844 IC50 = 66 nM T79031 CA4B6D 122196026 IC50 = 257 nM T79031 CEWY46 122196027 IC50 = 1445 nM T79031 C62JEW 122196028 IC50 = 5.2 nM T79031 C53POD 122196029 IC50 = 3.3 nM T79031 C2R6SY 122197438 IC50 = 550 nM T79031 CDG6R0 122197443 IC50 = 84 nM T79031 CG8H6M 122435134 Ki = 2.6 nM T79031 CIFT47 122484483 IC50 = 0.385 nM T79031 C35XVL 122535397 Ki = 26 nM T79031 CGLX79 122653795 IC50 = 0.157 nM T79031 CV7H1K 122660238 IC50 = 9.5 nM T79031 C1E3AZ 122660239 IC50 = 12 nM T79031 C52TCB 122660240 IC50 = 694 nM T79031 COW3Q1 122660243 IC50 = 9.5 nM T79031 CQNX38 122660245 IC50 = 21 nM T79031 C0AUG2 122660246 IC50 = 9 nM T79031 CAEX07 122662211 IC50 = 1 nM T79031 CO9J3K 122662227 IC50 = 2 nM T79031 CHM98B 122662233 IC50 = 1.5 nM T79031 CK7W8B 123132907 IC50 = 18 nM T79031 CRW0C2 123132915 IC50 = 0.024 nM T79031 CRMG32 126591378 Ki = 11 nM T79031 C45OVL 126693206 IC50 = 1.1 nM T79031 C1E7IG 126693231 IC50 = 1.2 nM T79031 CUF68P 126961340 EC50 = 18.5 nM T79031 CQ63PD 127025624 IC50 = 6040 nM T79031 C7M2LI 127025625 IC50 = 1000 nM T79031 CJT62C 127025626 IC50 = 730 nM T79031 CY53OH 127027133 IC50 = 2500 nM T79031 CMB8H5 127027134 IC50 = 140 nM T79031 CDG0C4 127027135 IC50 = 2280 nM T79031 C6N0XM 127027136 IC50 = 2690 nM T79031 CN50FI 127027450 IC50 = 40 nM T79031 C0Q7EF 127027451 IC50 = 400 nM T79031 CTB46J 127027772 IC50 = 390 nM T79031 C8TQ2G 127027773 IC50 = 1040 nM T79031 CBQ4E1 127027774 IC50 = 1080 nM T79031 C07GWU 127036055 IC50 = 430 nM T79031 CS6ND0 127036233 IC50 = 190 nM T79031 CT9E1M 127037187 IC50 = 6423 nM T79031 CH63BP 127037241 IC50 = 620 nM T79031 C39WGE 127038312 IC50 = 190 nM T79031 CG1K5J 127042875 IC50 = 600 nM T79031 CN84KA 127042876 IC50 = 210 nM T79031 C7S2LA 127044941 IC50 = 28 nM T79031 CS3Z7A 127045094 IC50 = 14 nM T79031 CSA71L 127046889 Ki = 57 nM T79031 CI9E4Q 127048180 IC50 = 31 nM T79031 CQ4ZF7 127048527 IC50 = 0.7 nM T79031 C7ON9C 127048528 IC50 = 2.3 nM T79031 C50OYT 127048529 IC50 = 160 nM T79031 C84TQV 127048530 IC50 = 0.7 nM T79031 CBU0D5 127050883 IC50 = 690 nM T79031 CN3XU0 127255875 IC50 = 22.2 nM T79031 CY1NE5 129011631 IC50 > 50000 nM T79031 C3MAO2 129011640 IC50 > 50000 nM T79031 CIK56O 129201653 Ki = 126 nM T79031 C4IQ6F 129201655 Ki = 42 nM T79031 CH5V3A 129201660 Ki = 4 nM T79031 C5Q1GT 129202050 Ki = 4 nM T79031 C19KGT 129202057 Ki = 10 nM T79031 CCBV68 129202062 Ki = 3 nM T79031 C7H3QJ 129202063 Ki = 22 nM T79031 CVMY58 129202069 Ki = 4 nM T79031 CLH8Z9 129202106 Ki = 23 nM T79031 CV78UP 132054712 IC50 = 2 nM T79031 CO63CX 132054802 IC50 = 4.8 nM T79031 CX27OU 132054828 IC50 = 0.9 nM T79031 CRJA89 132054902 IC50 = 7 nM T79031 C4UH5R 132054950 IC50 = 0.91 nM T79031 C4Y5UQ 132055484 Ki = 21 nM T79031 CD7AZ2 132068809 IC50 = 3.4 nM T79031 CEMC20 132230928 IC50 = 182 nM T79031 CLH6T3 132547257 IC50 = 16730 nM T79031 CXR7J9 132604796 IC50 = 15.5 nM T79031 CW0DO7 133703490 IC50 = 30300 nM T79031 C5T3YL 134130755 IC50 > 50000 nM T79031 CC5LZ6 134130905 IC50 = 20750 nM T79031 CGM75A 134131775 IC50 = 33 nM T79031 CU60NJ 134133911 IC50 = 600 nM T79031 COMC12 134141814 IC50 = 2000 nM T79031 CCM75O 134149181 IC50 = 82000 nM T79031 C0RKL4 134156261 IC50 = 230 nM T79031 CMA13L 134284187 IC50 = 8.18 nM T79031 CG8X9M 134822016 IC50 > 200000 nM T79031 C9W6JQ 135125856 IC50 = 1 nM T79031 CKVF19 135126469 IC50 = 8 nM T79031 CS06EN 135219058 IC50 = 49 nM T79031 C9ZYS8 135403573 IC50 = 28600 nM T79031 CS9G1Z 135416514 IC50 = 3000 nM T79031 C1WT4D 135424789 IC50 = 86000 nM T79031 CLC4O6 135436087 IC50 = 27200 nM T79031 CG5X9R 135492826 IC50 = 22000 nM T79031 CVD7Y3 135556691 IC50 = 2490000 nM T79031 CW81UQ 135566781 IC50 = 750 nM T79031 CC3QB7 135566786 IC50 = 470 nM T79031 CD39MX 135566787 IC50 = 170 nM T79031 C8TQ1R 135595416 IC50 = 2700 nM T79031 CAOL70 135875803 IC50 = 11000 nM T79031 CEZ79H 135875804 IC50 = 8000 nM T79031 CI1D7K 135875806 IC50 = 8200 nM T79031 CU0SF9 135875807 IC50 = 4600 nM T79031 C6J1EQ 135875808 IC50 = 110 nM T79031 CAT2H7 135875881 IC50 > 100000 nM T79031 CZY38L 135875883 IC50 > 100000 nM T79031 CYCA64 135875884 IC50 > 100000 nM T79031 CYD2F0 135887070 IC50 = 4800 nM T79031 CUXV05 135960747 IC50 > 100000 nM T79031 CQT02Z 135985898 IC50 = 130 nM T79031 C2WYV6 135998870 IC50 > 100000 nM T79031 C1VZN5 136016387 IC50 = 500000 nM T79031 CKRG38 136016388 IC50 = 100000 nM T79031 C9R3GS 136016426 IC50 = 100000 nM T79031 C32HVK 136078846 IC50 > 160000 nM T79031 CWY19J 136086725 IC50 = 7.9 nM T79031 CL0R8V 136086726 IC50 = 10 nM T79031 CFHQ58 136094849 IC50 = 6.6 nM T79031 CT0N8B 136219145 IC50 = 590 nM T79031 C7NQZ1 136219146 IC50 = 73700 nM T79031 C7XNV5 136219147 IC50 = 560 nM T79031 CW1ZL7 136219148 IC50 = 7230 nM T79031 CN71UO 136219149 IC50 = 2710 nM T79031 C2JO1Y 136219150 IC50 = 3370 nM T79031 CNY56O 136219151 IC50 > 250000 nM T79031 CU8VW3 136219152 IC50 = 137100 nM T79031 C9R1ED 136219153 IC50 = 339700 nM T79031 CB7L6W 136219154 IC50 = 184900 nM T79031 CI89QA 136219155 IC50 = 638600 nM T79031 C0QUP1 136219156 IC50 = 2840 nM T79031 CQ1A5E 136219157 IC50 = 5410 nM T79031 CD3RK6 136219248 IC50 = 310 nM T79031 C3T2FQ 136219249 IC50 = 9500 nM T79031 C6QEC7 136219250 IC50 = 1260 nM T79031 CK3R8X 136219251 IC50 = 8 nM T79031 C60STM 136219252 IC50 = 406 nM T79031 C2FDN6 136229320 IC50 = 2900 nM T79031 CQ4E3V 136229321 IC50 = 710 nM T79031 CH1C8U 136229322 IC50 = 1850 nM T79031 C20DYZ 136229323 IC50 = 820 nM T79031 CW7VZ2 136229324 IC50 = 450 nM T79031 CAFC51 136229325 IC50 = 1090 nM T79031 C5V9IE 136229326 IC50 = 630 nM T79031 CTX80B 136229327 IC50 = 610 nM T79031 C2R6UH 136229328 IC50 = 570 nM T79031 C14DGV 136229329 IC50 = 2430 nM T79031 C35QWB 136229330 IC50 = 760 nM T79031 CAS8G6 136229331 IC50 = 510 nM T79031 CR2YQ0 136236289 IC50 = 130000 nM T79031 CV0Q6S 136239432 IC50 = 263800 nM T79031 CV0Y1W 136266507 Ki = 2.8 nM T79031 C8L5PZ 137348437 IC50 = 0.62 nM T79031 CLE04H 137348743 IC50 = 0.31 nM T79031 CYLI20 137392390 IC50 = 0.09 nM T79031 CES5F6 137462330 Ki = 1.9 nM T79031 CCW43D 137631772 Ki = 23 nM T79031 CY2J3K 137632461 IC50 = 6840 nM T79031 C8P1CN 137632526 Ki = 22200 nM T79031 C8JWF7 137633017 IC50 = 5890 nM T79031 CD15MW 137633338 IC50 = 310 nM T79031 CG5C1T 137634151 IC50 = 5 nM T79031 CU40QT 137634377 IC50 = 12 nM T79031 CLK7A3 137635011 IC50 = 64 nM T79031 CY5M8Z 137635828 IC50 = 53 nM T79031 CIV59G 137636278 Ki = 320 nM T79031 C6RIC3 137636763 Ki = 300 nM T79031 CET5V4 137637305 IC50 = 530 nM T79031 CE2WL0 137637333 IC50 = 110 nM T79031 C2B1MZ 137637375 IC50 = 14 nM T79031 CL80TF 137637682 IC50 = 1670 nM T79031 CEVA49 137637780 IC50 = 8 nM T79031 CTB58M 137638219 EC50 = 590 nM T79031 C7CE1X 137638268 IC50 = 21 nM T79031 CB09LG 137638295 IC50 = 4900 nM T79031 CXG42C 137638912 IC50 = 1.1 nM T79031 CSQL63 137640486 IC50 = 38 nM T79031 CKC6N9 137641085 IC50 = 7 nM T79031 CR8TY4 137641223 IC50 = 130 nM T79031 C91GMY 137641491 IC50 = 30 nM T79031 COD81X 137642018 IC50 = 1.05 nM T79031 CM6G4J 137642066 Ki = 175.5 nM T79031 C63QPE 137642336 IC50 = 480 nM T79031 CTYP90 137642839 IC50 = 1500 nM T79031 C9BF0V 137643369 IC50 = 60 nM T79031 C0BM2P 137644926 Ki = 20.5 nM T79031 CV56QL 137645221 IC50 = 17 nM T79031 CG3U5K 137645264 Ki = 2 nM T79031 C9OV2Q 137646113 IC50 = 2.7 nM T79031 CTB27V 137646126 IC50 = 4 nM T79031 C10CBD 137646316 IC50 = 400 nM T79031 CLF8P5 137646591 IC50 = 1.5 nM T79031 CJXK40 137648425 IC50 = 2 nM T79031 CL2O7F 137648801 IC50 = 99 nM T79031 C6JO1R 137649130 IC50 = 114.8 nM T79031 C51XRG 137650311 Ki = 26 nM T79031 CM24RN 137650832 Ki = 144 nM T79031 CTKL23 137651107 IC50 = 85 nM T79031 C6P8IL 137651254 IC50 = 120 nM T79031 CVR29E 137651451 IC50 = 24 nM T79031 C97CST 137651879 IC50 > 200000 nM T79031 C8HSX7 137652983 IC50 = 8200 nM T79031 CL3DW0 137653017 IC50 = 5.9 nM T79031 CMH21N 137653098 IC50 = 2600 nM T79031 CJB10E 137653201 Ki = 12 nM T79031 CQ32NO 137653545 IC50 = 490 nM T79031 CBE82Q 137653962 IC50 = 212 nM T79031 CL7W9I 137653970 EC50 = 480 nM T79031 CS7UO6 137654080 Ki = 32600 nM T79031 CK3F9G 137654547 IC50 = 180 nM T79031 CXY7F1 137654633 IC50 = 73500 nM T79031 CQ9T6V 137655111 IC50 = 98 nM T79031 C5LPG4 137655356 IC50 = 800 nM T79031 CTU5C1 137656577 IC50 = 4 nM T79031 CJ8WD4 137657298 Ki = 5690 nM T79031 C3L8WX 137657646 IC50 = 20200 nM T79031 C1ULD3 137660988 IC50 = 2.9 nM T79031 C3YFL4 137662127 IC50 = 22 nM T79031 C7U4IN 137662155 IC50 = 75 nM T79031 C1MRT7 138454796 Ki = 1.9 nM T79031 CXU9Y2 138459258 IC50 = 2 nM T79031 C8DH9F 138857908 IC50 = 1.7 nM T79031 CE35GB 138857909 IC50 = 2 nM T79031 CEG59N 139590110 IC50 > 50000 nM T79031 C7VPS5 139590111 IC50 > 50000 nM T79031 CPUI86 139590112 IC50 = 3320 nM T79031 CQK1J0 139590113 IC50 = 5850 nM T79031 CCI39R 139590114 IC50 > 50000 nM T79031 CGQ6T2 139590115 IC50 > 50000 nM T79031 C4L0DZ 139590116 IC50 > 50000 nM T79031 CQ8KC9 139590117 IC50 = 31680 nM T79031 CS06KY 139590118 IC50 > 50000 nM T79031 CX8GT9 139590119 IC50 > 50000 nM T79031 C48XFW 142342111 IC50 = 1.86 nM T79031 CC4T3Y 145949506 IC50 = 40.3 nM T79031 CDL20Q 145950148 IC50 = 6400 nM T79031 CF43XD 145951346 IC50 = 3020 nM T79031 CR25WD 145951471 IC50 = 4400 nM T79031 CP19IT 145952557 IC50 = 30.2 nM T79031 C4T8GH 145952957 IC50 = 24.5 nM T79031 C06AYZ 145953144 IC50 = 41400 nM T79031 C8P5CU 145953623 IC50 = 2200 nM T79031 CB6O5F 145953952 IC50 = 106700 nM T79031 CSN91F 145953996 IC50 = 11 nM T79031 CE6CT0 145954147 IC50 = 6.4 nM T79031 C2D1CW 145954300 IC50 = 7500 nM T79031 C9D4GK 145954965 IC50 = 18500 nM T79031 C82RDB 145955110 IC50 = 35.1 nM T79031 CT5AX1 145955169 IC50 = 19100 nM T79031 CP3RZ8 145955538 IC50 = 2200 nM T79031 C4T8AB 145955939 IC50 = 1862 nM T79031 CK5CL0 145956622 IC50 = 40.7 nM T79031 CBT43H 145957650 IC50 = 115 nM T79031 C0OFL6 145957885 IC50 = 6800 nM T79031 CGO35N 145959085 IC50 = 15600 nM T79031 CP7KE9 145959864 IC50 = 1700 nM T79031 C4MDJ7 145960187 IC50 = 10.7 nM T79031 CB5O9V 145960446 IC50 = 38 nM T79031 C7NBQ6 145960692 IC50 = 3200 nM T79031 C45TMN 145960757 Ki = 206 nM T79031 C98AVO 145960781 IC50 = 4500 nM T79031 CI3C4K 145960897 IC50 = 38600 nM T79031 CZ83AF 145960980 IC50 = 27600 nM T79031 C0D6OX 145961033 IC50 = 53 nM T79031 CPFG08 145961278 IC50 = 29600 nM T79031 CRA4L0 145961341 IC50 = 37400 nM T79031 C8UHR3 145961471 IC50 = 26100 nM T79031 C41MDH 145961476 IC50 = 26 nM T79031 C1KMU8 145961539 Ki = 4 nM T79031 CVQM71 145961719 IC50 = 24300 nM T79031 CF3H9W 145961985 IC50 = 7700 nM T79031 CS3MR2 145962254 IC50 = 15000 nM T79031 C6E7LS 145962264 IC50 = 69 nM T79031 CO6J8R 145962333 IC50 = 17500 nM T79031 CYV2M3 145962371 IC50 = 13500 nM T79031 CZ70SW 145962377 IC50 = 4200 nM T79031 COI9X0 145962778 Ki = 36 nM T79031 C5MOA0 145962826 IC50 = 25 nM T79031 CVU70C 145962834 Ki = 31 nM T79031 CVH8K9 145963013 IC50 = 13400 nM T79031 C7BY9K 145963167 IC50 = 4 nM T79031 CMN62K 145963255 IC50 = 15000 nM T79031 C6ZXY4 145963432 IC50 = 1077 nM T79031 CR7J6S 145963458 IC50 = 663 nM T79031 CL49ZJ 145963489 IC50 = 27 nM T79031 C0G6IC 145963607 IC50 = 4600 nM T79031 CNG5K7 145964592 IC50 = 1700 nM T79031 CDZS20 145964643 IC50 > 50000 nM T79031 CTD64W 145964995 Ki = 2.74 nM T79031 C8XS9J 145965252 IC50 = 2500 nM T79031 CJP34X 145965420 IC50 = 6060 nM T79031 C1J5ZO 145965555 Ki = 2.14 nM T79031 CCF43R 145965575 Ki = 4.59 nM T79031 CDO2Q5 145965821 IC50 > 50000 nM T79031 CG1EQ2 145965859 IC50 > 10000 nM T79031 C36CZY 145966369 IC50 = 2920 nM T79031 CNQT09 145966611 Ki = 209.27 nM T79031 CN69LR 145966948 IC50 = 6500 nM T79031 C3FP4K 145967185 Ki = 2.62 nM T79031 C0H5UD 145967429 IC50 = 0.033 nM T79031 C1S2WH 145968008 IC50 = 4100 nM T79031 CP2L3Q 145969138 IC50 = 2400 nM T79031 CL05SA 145969593 IC50 = 2800 nM T79031 CE8RJ4 145970093 IC50 > 10000 nM T79031 C5DGW7 145970482 IC50 = 2700 nM T79031 CP6ET4 145971201 IC50 = 12.2 nM T79031 CGKQ14 145971440 IC50 = 251 nM T79031 C2OBD4 145971568 Ki = 2.77 nM T79031 C53OSI 145971666 IC50 = 0.034 nM T79031 C64PUZ 145972542 IC50 > 10000 nM T79031 CN5Z4D 145973319 IC50 = 3200 nM T79031 CRVP34 145973792 Ki = 31.17 nM T79031 C8F7AM 145974484 Ki = 10.33 nM T79031 CVK1O7 145974594 IC50 = 250 nM T79031 CVM02B 145974600 IC50 = 2050 nM T79031 CTS45U 145974623 Ki = 4.38 nM T79031 C3S2ON 145975161 IC50 > 50000 nM T79031 C38FJD 145975195 IC50 = 3000 nM T79031 C0GN1C 145975379 IC50 = 1600 nM T79031 CJD54C 145975664 Ki = 104.73 nM T79031 CG4IV1 145976106 IC50 = 11 nM T79031 CR48PN 145976179 Ki = 20.13 nM T79031 CJ7T1L 145976222 Ki = 5.03 nM T79031 CQ1MO0 145976476 IC50 = 3600 nM T79031 C8ZLF2 145976856 Ki = 4.46 nM T79031 CKU21C 145977020 IC50 = 5170 nM T79031 CM27YI 145977049 IC50 = 110 nM T79031 CX1R7K 145977083 Ki = 14.67 nM T79031 CCI94W 145977228 IC50 = 1900 nM T79031 C49DPO 145977509 Ki = 1.37 nM T79031 CO0G5I 145978024 IC50 = 3800 nM T79031 C0H6IP 145978056 IC50 = 5700 nM T79031 CYH46T 145978250 IC50 = 0.11 nM T79031 CHJ2N9 145978340 IC50 = 3800 nM T79031 CVK9J5 145978628 IC50 = 1330 nM T79031 C7DH9J 145979410 IC50 = 4000 nM T79031 CZX3G9 145979423 IC50 = 5000 nM T79031 C01PMA 145979438 Ki = 1 nM T79031 CD6C2Q 145979768 IC50 = 2100 nM T79031 C2D5YT 145980015 Ki = 1 nM T79031 CI4C2V 145980078 IC50 = 5.5 nM T79031 CGQO25 145980230 IC50 = 1600 nM T79031 CV6N5E 145980299 IC50 = 3.6 nM T79031 CL2O0B 145980889 IC50 = 1.8 nM T79031 C2WVP9 145980947 IC50 = 2600 nM T79031 C3BS5J 145981023 IC50 = 13 nM T79031 CB7LD6 145981185 Ki = 1 nM T79031 C79EQW 145981356 Ki = 100 nM T79031 CA0Y1X 145981628 Ki = 1 nM T79031 C1Y3NM 145981718 IC50 = 2000 nM T79031 C3OD9P 145981738 IC50 = 1200 nM T79031 CLG9V4 145982062 Ki = 1 nM T79031 CJV1E8 145983023 Ki = 4124 nM T79031 CE8G4K 145983065 Ki = 41126 nM T79031 CBA5F1 145983114 Ki = 110.5 nM T79031 CQ6F2O 145983136 Ki = 630 nM T79031 C4XG5A 145983198 IC50 = 0.46 nM T79031 C17GWT 145983210 IC50 = 72 nM T79031 C5QUR7 145983971 Ki = 28758 nM T79031 CFR8V0 145984198 Ki = 553.7 nM T79031 C48AJL 145984450 Ki = 28.1 nM T79031 COJ41C 145985693 Ki = 10.9 nM T79031 CA27NB 145986108 Ki = 808.6 nM T79031 CWP2Q5 145986616 IC50 = 31 nM T79031 CV6R9D 145986652 IC50 = 1600 nM T79031 CTL5Y0 145986900 Ki = 10 nM T79031 CIE06B 145987057 IC50 = 2800 nM T79031 COB69L 145987073 Ki = 0.7 nM T79031 CK9L8J 145987341 IC50 = 0.58 nM T79031 C91UHM 145988149 IC50 = 3600 nM T79031 CMP51W 145988521 IC50 = 2600 nM T79031 CVD20U 145988532 IC50 > 10000 nM T79031 C68NKP 145988628 IC50 = 83.6 nM T79031 CNC1H3 145988728 IC50 = 190 nM T79031 CY57HJ 145988915 IC50 = 1200 nM T79031 CK2GE9 145989033 IC50 = 71.5 nM T79031 CI96PW 145989240 IC50 = 1700 nM T79031 C70HDR 145989886 Ki = 0.7 nM T79031 C6QRA9 145989946 IC50 > 10000 nM T79031 CTJ5L4 145989961 IC50 > 10000 nM T79031 C8RGA4 145990244 Ki = 4 nM T79031 CUGP43 145990468 IC50 = 0.43 nM T79031 CZK41W 145990916 IC50 = 7.5 nM T79031 CN7I8T 145991278 IC50 = 0.92 nM T79031 C1ZQ0W 145991508 IC50 > 10000 nM T79031 CSAI70 145991785 IC50 = 0.57 nM T79031 C0KNI4 145991888 Ki = 2 nM T79031 C57CEQ 145991917 IC50 = 2800 nM T79031 CG9WR4 145991995 IC50 = 4300 nM T79031 C0QI3G 145992571 IC50 = 2000 nM T79031 C3PD7L 145992760 Ki = 1 nM T79031 CA1QE7 145993306 Ki = 3 nM T79031 CY2N1D 145993326 IC50 > 10000 nM T79031 CH3EP0 145993573 Ki = 10 nM T79031 C1RPM8 145993657 IC50 = 2100 nM T79031 CY37RJ 145994215 Ki = 1 nM T79031 CP5Y4L 146737289 IC50 = 1300 nM T79031 CKB5X0 148667961 IC50 = 1800 nM T79031 C06MWU 148980171 IC50 = 1100 nM T79031 CRKM38 149207555 IC50 = 3600 nM T79031 CYTQ79 153303564 IC50 = 9.6 nM T79031 CBC6S2 154031826 IC50 = 3 nM T79031 C83RXG 154031827 IC50 = 22.91 nM T79031 C65UKV 155510422 IC50 = 3162.28 nM T79031 C0GU8Q 155510649 IC50 = 328.1 nM T79031 CRD8I0 155510888 IC50 > 10000 nM T79031 CILH15 155512503 IC50 = 30 nM T79031 CY6Q9U 155512597 IC50 = 5.4 nM T79031 C23BDU 155512711 IC50 = 180 nM T79031 CM7U1J 155513259 IC50 = 6.026 nM T79031 CL53YZ 155513311 IC50 = 6.23 nM T79031 CY0E3D 155514519 IC50 = 14000 nM T79031 CR7C0G 155515606 IC50 = 2400 nM T79031 C7V8ZP 155516667 Ki = 4 nM T79031 CR4P3Z 155516698 IC50 = 2900 nM T79031 CHVY37 155516817 IC50 = 1109 nM T79031 C28AKI 155517345 IC50 = 970 nM T79031 CU9B6X 155517833 IC50 = 5.67 nM T79031 C3NMX4 155517840 IC50 = 220.4 nM T79031 CSU3P7 155518836 IC50 = 97.72 nM T79031 C6J9RB 155520405 IC50 = 320 nM T79031 C1H7YT 155520705 IC50 = 11.2 nM T79031 CZR0D3 155520717 IC50 = 1800 nM T79031 CJE93X 155520921 IC50 = 22 nM T79031 CGK13P 155521616 IC50 > 10000 nM T79031 CHG5D0 155521756 IC50 = 730 nM T79031 CKO59Y 155522051 IC50 = 4.5 nM T79031 C34RWB 155522578 IC50 > 10000 nM T79031 C43GKJ 155522872 IC50 = 456.2 nM T79031 CAGO28 155523111 IC50 > 10000 nM T79031 CEW74K 155523671 IC50 = 420 nM T79031 CS6IJ2 155524198 IC50 = 12000 nM T79031 C40DMT 155526564 Ki = 9.1 nM T79031 CUY0L8 155528391 IC50 = 1.6 nM T79031 CCWA24 155529695 IC50 = 720.5 nM T79031 C4FLZ0 155530158 IC50 = 7079 nM T79031 CEH06J 155530168 IC50 = 173.5 nM T79031 C54GFT 155532930 IC50 > 10000 nM T79031 CP8EX6 155535061 IC50 > 10000 nM T79031 COW05C 155536534 Ki = 3 nM T79031 CVA2L3 155536581 IC50 = 141.4 nM T79031 CKGP95 155536618 IC50 = 6.607 nM T79031 CL53AK 155537567 IC50 > 10000 nM T79031 COF63Z 155537873 IC50 = 6.13 nM T79031 CUK21B 155538074 IC50 = 1.3 nM T79031 CME8I2 155538181 IC50 > 10000 nM T79031 C2B5ID 155538495 Ki = 22 nM T79031 C1W7DO 155538806 IC50 = 0.95 nM T79031 CKGC96 155538886 IC50 > 10000 nM T79031 CY9NM8 155539369 IC50 = 3700 nM T79031 CF6E1H 155539416 IC50 > 10000 nM T79031 C0BQ9M 155540237 IC50 = 55200 nM T79031 CC9YP3 155540604 IC50 = 33884.42 nM T79031 CFW15C 155540816 IC50 > 10000 nM T79031 CI64ZO 155541480 IC50 = 1500 nM T79031 CTKH05 155541830 IC50 = 30.9 nM T79031 C2MOI5 155541886 IC50 > 10000 nM T79031 C5Q7LX 155542202 IC50 = 84000 nM T79031 C4TQN1 155542315 IC50 = 5.888 nM T79031 CB9V1D 155543145 Ki = 22 nM T79031 CL9Z6H 155543895 IC50 > 10000 nM T79031 C17JEA 155543947 IC50 = 18400 nM T79031 CV4MO2 155544490 IC50 = 1700 nM T79031 CG28VK 155544704 IC50 = 300 nM T79031 CF6XZ8 155544727 IC50 = 1.6 nM T79031 CI51DC 155547003 IC50 = 119.4 nM T79031 C65EWF 155547684 IC50 = 172 nM T79031 C6PI3K 155547763 IC50 = 14700 nM T79031 CD8JZ5 155548223 IC50 = 3400 nM T79031 C14SPW 155548636 IC50 > 10000 nM T79031 CPHJ28 155548834 IC50 = 10.23 nM T79031 CMA98V 155548892 IC50 = 49800 nM T79031 CVS8G7 155549034 IC50 = 1047 nM T79031 CV8PL5 155549546 IC50 = 851.2 nM T79031 C79KNV 155550335 IC50 = 195.3 nM T79031 CP86OC 155551378 IC50 = 230 nM T79031 CBG0E9 155552470 IC50 = 1575 nM T79031 CP90YG 155553358 IC50 = 424.9 nM T79031 C0DX5G 155553529 IC50 = 54954.09 nM T79031 CS32WZ 155553812 IC50 = 11400 nM T79031 COG0L9 155553890 IC50 = 8550 nM T79031 CMXP34 155555473 IC50 = 420 nM T79031 CMK57Q 155556223 IC50 = 410 nM T79031 CQ2J3F 155556725 IC50 = 6.9 nM T79031 C7S5JN 155556840 IC50 = 10000 nM T79031 CYF36J 155557043 IC50 = 11420 nM T79031 CW3E7A 155557894 IC50 = 33000 nM T79031 CHN4S6 155558787 IC50 = 4.77 nM T79031 CLYI80 155559529 IC50 = 7.2 nM T79031 C62BUJ 155560190 IC50 = 34000 nM T79031 C0SQ7I 155560420 IC50 = 3900 nM T79031 C2KUE9 155560600 IC50 = 1.8 nM T79031 CI8UF7 155560617 IC50 = 3500 nM T79031 CLY7Q6 155560920 IC50 = 19000 nM T79031 C95CBX 155561050 IC50 = 280 nM T79031 CP7I9L 155561118 IC50 = 3300 nM T79031 C5BU7H 155561129 IC50 = 480 nM T79031 C6RXE2 155561338 IC50 = 6100 nM T79031 C9QG3Y 155562174 IC50 = 77.62 nM T79031 CNQ9D5 155563009 IC50 = 5100 nM T79031 CM2QK1 155563180 IC50 > 10000 nM T79031 C6DKB9 155563223 IC50 = 0.99 nM T79031 C7BCO6 155563658 IC50 = 1.1 nM T79031 C4QX9B 155565034 IC50 = 2691.53 nM T79031 CBS97E 155565975 Ki = 6.5 nM T79031 C7TK8V 155566239 IC50 = 20.7 nM T79031 C7NJY2 155566392 IC50 = 1400 nM T79031 C93SNX 155566643 IC50 = 2 nM T79031 CL14DJ 155566956 IC50 = 160 nM T79031 C6Z2SM 155567115 IC50 = 28840.32 nM T79031 C2Z0TE 155567198 IC50 = 86700 nM T79031 CA8T0P 155567230 IC50 = 0.2 nM T79031 CBX2E3 155567555 IC50 > 10000 nM T79031 C4X7OL 155567906 IC50 = 250 nM T79031 C0QJL4 155568510 IC50 = 1.03 nM T79031 C3C1XH 11497497 IC50 = 93 nM T79031 CBQP67 11613166 IC50 = 12 nM T79031 C1KYA7 46877606 IC50 = 14 nM T79031 D00CYX 44397266 Ki = 0.3 nM T79031 D00QDR 65238 IC50 = 3760 nM T79031 D00RIX 5280443 IC50 = 38500 nM T79031 D00SDQ 50938551 IC50 = 0.84 nM T79031 D02AQM 6918822 IC50 = 1600 nM T79031 D02JEZ 5281426 IC50 > 500000 nM T79031 D02LCH 16659106 Ki = 1.1 nM T79031 D03VQF 11982641 IC50 = 6700 nM T79031 D03ZMQ 323 IC50 > 500000 nM T79031 D04RSC 447068 Ki = 0.3 nM T79031 D07EWF 66575082 Ki = 1.7 nM T79031 D07KXK 5276890 Ki = 170 nM T79031 D08ALW 449218 Ki = 25 nM T79031 D08HZD 11701820 IC50 = 100000 nM T79031 D08MZY 145937 IC50 = 12200 nM T79031 D08UYP 3008868 Ki = 1500 nM T79031 D09ROW 10212 IC50 = 30500 nM T79031 D09SOY 15054176 EC50 = 3400 nM T79031 D0A0RO 10397869 IC50 = 310000 nM T79031 D0A1CM 5281855 IC50 = 3900 nM T79031 D0C1LI 53378764 IC50 = 460 nM T79031 D0D4FV 44593449 Ki = 3900 nM T79031 D0D5YP 5280371 IC50 > 500000 nM T79031 D0F3QP 5889042 IC50 = 9800 nM T79031 D0G3TK 5280863 IC50 = 14700 nM T79031 D0H0SE 21626545 IC50 = 11680 nM T79031 D0H3EJ 11205295 IC50 = 16 nM T79031 D0I8KC 11586735 IC50 = 94000 nM T79031 D0K2XJ 442679 IC50 = 3100 nM T79031 D0L7AT 10480940 Ki = 7200 nM T79031 D0M4IE 9549196 IC50 = 7500 nM T79031 D0NJ4H 5281670 IC50 = 12300 nM T79031 D0O0FA 44563121 IC50 = 2600 nM T79031 D0O0GW 71202307 IC50 = 26 nM T79031 D0RB1V 6419835 IC50 = 6000 nM T79031 D0S0BN 130976 Ki = 1300 nM T79031 D0S1MC 23643351 IC50 = 238 nM T79031 D0T3PW 5281672 IC50 = 2800 nM T79031 D0U4BB 10748 IC50 > 500000 nM T79031 D0VE0Q 72936 Ki = 1100 nM T79031 D0W4ZU 44563198 IC50 = 39200 nM T79031 D0WA9S 10429214 IC50 = 5350 nM T79031 D0Y5IQ 44255320 IC50 = 10000 nM T79031 D0YZ5G 5281416 IC50 > 500000 nM T19492 D0K9IF 71666749 IC50 > 30000 nM T19492 C6HA8E 5388709 IC50 > 30000 nM T19492 C8W2QA 6439099 IC50 > 30000 nM T19492 C8NM2I 11538313 EC50 = 10000 nM T19492 CA5W9R 11618060 EC50 = 1400 nM T19492 CLT3Z7 11695929 EC50 = 2500 nM T19492 CQSZ72 90675942 IC50 > 30000 nM T19492 CTBD74 90675943 IC50 > 30000 nM T19492 CM12LR 102597975 IC50 > 30000 nM T19492 CW9P6A 145964460 IC50 > 30000 nM T19492 CQR49Z 145965116 IC50 > 30000 nM T19492 CR6L2G 145967358 IC50 > 30000 nM T19492 CHXE25 145978207 IC50 > 30000 nM T19492 D08BMM 6312649 IC50 = 20000 nM T19492 D0R9CF 11302540 IC50 = 450 nM T67339 CM15EI 23582895 Ki = 12 nM T67339 CA9H3O 44563619 Ki > 100000 nM T67339 CF2RI5 44563620 Ki > 100000 nM T67339 C5LTM8 44563621 Ki = 15200 nM T67339 CAB72K 44563622 Ki = 5720 nM T67339 CK3MA7 44563623 Ki = 5780 nM T67339 CLEV46 44563624 Ki = 2100 nM T67339 CAV6L7 44563625 Ki = 1400 nM T67339 C89VHR 44563626 Ki = 267 nM T67339 CVQH25 44563627 Ki = 49 nM T67339 C78YXV 44563628 Ki = 40 nM T67339 C2F3VC 44563629 Ki = 1040 nM T67339 CEL16A 44563630 Ki = 41 nM T67339 CP91ZQ 44563631 Ki = 28 nM T67339 CIH2P9 44563632 Ki = 45 nM T67339 C1D6RW 44563633 Ki = 27 nM T67339 C8WMU0 44563634 Ki = 19 nM T67339 C8AMN7 44563635 Ki = 65 nM T67339 CGH2L9 44563636 Ki = 130 nM T67339 C4Z6VO 44563637 Ki = 60 nM T67339 C6J0QY 44563638 Ki = 176 nM T67339 CQGT25 44563639 Ki = 29 nM T67339 C2Z7DI 44563640 Ki = 101 nM T67339 C9Q0PG 44563641 Ki = 510 nM T67339 CY59RO 44563642 Ki = 1550 nM T13852 D07UHS 107970 EC50 = 0.3 nM T13852 D07EDB 52938427 EC50 = 0.16 nM T13852 D07FKQ 44599207 EC50 = 0.4 nM T13852 D07UGA 5283560 EC50 = 0.027 nM T13852 D0HI1K 107969 EC50 = 3000 nM T13852 D0I2RB 11502996 EC50 = 0.027 nM T13852 D0L9KH 44623998 EC50 = 0.04 nM T13852 D0Y4SI 11363176 EC50 = 9.7 nM T13852 D04NEO 25031140 EC50 = 0.2 nM T13852 D04UXN 25182901 EC50 = 6 nM T13852 D09LDU 25182746 EC50 = 390 nM T13852 D0EP8Y 86299710 EC50 = 5.1 nM T13852 D0HW8T 76325532 EC50 = 0.2 nM T13852 D0I5TH 25182905 EC50 = 36 nM T13852 D0K4BI 10223146 IC50 > 1000 nM T13852 D0LT2N 25182763 EC50 = 405 nM T13852 D0PW0R 71547555 IC50 > 10000 nM T13852 D0R7ED 76325522 EC50 = 0.1 nM T13852 C3RZ6P 904918 EC50 = 86 nM T13852 C1E4SA 1009742 EC50 = 430 nM T13852 CAXQ30 1160318 EC50 = 19952.62 nM T13852 C7QC0W 1776080 EC50 = 819 nM T13852 CPO6B9 2740144 IC50 = 25 nM T13852 CN29JD 2799937 IC50 = 27 nM T13852 CE2LQ9 3212803 EC50 = 199.53 nM T13852 CZ9UI1 3212804 EC50 = 1258.93 nM T13852 C4WI2Z 3212805 EC50 = 251.19 nM T13852 CS1PB7 3212808 EC50 = 794.33 nM T13852 C2HP3Z 3212809 EC50 = 630.96 nM T13852 C2ZH6U 3245758 EC50 > 50000 nM T13852 CRZ85P 3721977 EC50 = 1258.93 nM T13852 CT4M1V 3868087 EC50 = 6.7 nM T13852 C7N5UR 4107292 IC50 = 78 nM T13852 CPLQ54 4225876 EC50 = 31622.78 nM T13852 C5O6YL 4318239 EC50 = 1030 nM T13852 CIA43B 4492589 IC50 > 20000 nM T13852 CV69WH 5307570 EC50 > 50000 nM T13852 C89ATE 5309153 EC50 = 7870 nM T13852 CZE96X 6056442 IC50 = 6180 nM T13852 C2X9ZN 6857803 Ki = 2840 nM T13852 C72DNW 9796603 IC50 = 150 nM T13852 CS8MB9 9821227 EC50 = 12.7 nM T13852 C1K9GW 9824415 IC50 = 7.3 nM T13852 CW37CN 9969355 EC50 = 160 nM T13852 C7FGR9 9979368 IC50 = 1.4 nM T13852 CI3K9Z 10023913 EC50 = 8.6 nM T13852 CZLT30 10045980 IC50 = 2.9 nM T13852 CA4HX3 10125861 IC50 = 19 nM T13852 C8KXE2 10125862 IC50 = 22 nM T13852 CG6O1W 10125882 IC50 = 41 nM T13852 C7B8UT 10126584 IC50 = 0.3 nM T13852 CG65LQ 10126736 IC50 = 2.5 nM T13852 CN8H2S 10127475 EC50 = 0.5 nM T13852 CCG97S 10127776 IC50 = 4.1 nM T13852 CGCK28 10149985 IC50 = 0.2 nM T13852 CO06YT 10150171 IC50 = 0.76 nM T13852 C3LG4R 10150372 IC50 = 0.5 nM T13852 CPU38H 10151146 IC50 = 0.6 nM T13852 CE9WX6 10172338 IC50 = 8.4 nM T13852 CDE1S4 10172354 IC50 = 1.5 nM T13852 CI5X6K 10172513 IC50 = 0.9 nM T13852 CWJO04 10172546 IC50 = 0.3 nM T13852 CS62VA 10173002 IC50 = 2.3 nM T13852 CL2QV0 10173327 IC50 = 2.4 nM T13852 CSV6Q3 10174181 IC50 = 1.4 nM T13852 C5XFN7 10174255 EC50 = 0.2 nM T13852 C8XZV1 10174548 IC50 = 1.2 nM T13852 CG3DX8 10193676 IC50 = 44 nM T13852 CR9YM8 10193915 IC50 = 0.7 nM T13852 C5HJB9 10195325 EC50 = 2.4 nM T13852 CY1T7W 10215138 IC50 = 25 nM T13852 C56XBS 10215741 IC50 = 2.3 nM T13852 CN2FJ9 10216035 IC50 = 1600 nM T13852 C6NP8S 10217498 EC50 = 1.4 nM T13852 C9KH2F 10236683 IC50 = 7.7 nM T13852 CN93ZD 10249887 IC50 = 3.8 nM T13852 C6H9VI 10249979 IC50 = 1.8 nM T13852 C2O4UR 10251062 IC50 = 1.7 nM T13852 C2YZC3 10271422 IC50 = 6 nM T13852 CN0EC2 10286857 IC50 = 2 nM T13852 CKPV49 10287091 IC50 = 32 nM T13852 C74CKG 10287343 IC50 = 1.9 nM T13852 CW5JG7 10287365 IC50 = 0.9 nM T13852 C3R1AI 10288370 IC50 = 13 nM T13852 C5MDF6 10288527 EC50 = 0.8 nM T13852 C6EY2U 10289318 IC50 = 1.3 nM T13852 CJ26CW 10308738 IC50 = 14 nM T13852 C2U3LT 10309022 IC50 = 1700 nM T13852 C8VP3G 10309271 IC50 = 14 nM T13852 C7B2FU 10309462 IC50 = 0.4 nM T13852 CAF85E 10310253 IC50 = 0.4 nM T13852 CPK61C 10310952 IC50 = 33 nM T13852 C8HBY4 10311227 IC50 = 0.4 nM T13852 C3SM5Z 10317453 IC50 = 1.3 nM T13852 CG89DO 10363915 IC50 = 1.3 nM T13852 CDV3W7 10384596 IC50 = 0.1 nM T13852 C8WL6R 10408874 IC50 = 0.4 nM T13852 COQ65E 10409838 IC50 = 29 nM T13852 CI3EW1 10430549 IC50 = 0.6 nM T13852 CAL72D 10476387 IC50 = 3.8 nM T13852 C9NRD6 11168252 EC50 = 5.9 nM T13852 CZ3T0G 11177439 EC50 > 10000 nM T13852 CD8T1W 11222939 EC50 = 0.14 nM T13852 CUR1P8 11224984 EC50 = 5.7 nM T13852 CFPH94 11248292 EC50 = 1.3 nM T13852 CK65MP 11271470 EC50 = 1.4 nM T13852 C6N4UQ 11280849 EC50 = 11 nM T13852 CVJX85 11313781 EC50 = 70 nM T13852 C9JZP8 11315069 EC50 = 95 nM T13852 C34OBY 11315717 EC50 = 2.9 nM T13852 C6ZFY8 11315809 EC50 = 0.84 nM T13852 COS3Y2 11360553 EC50 = 45 nM T13852 CAS3N4 11371585 EC50 = 43 nM T13852 C6JX5O 11397995 EC50 = 0.7 nM T13852 C69NSZ 11405953 EC50 = 150 nM T13852 C9NOJ7 11406331 EC50 = 2400 nM T13852 CYH0U8 11408903 EC50 = 1.3 nM T13852 CER35T 11466640 EC50 = 3.3 nM T13852 C1SMT3 11484624 EC50 = 2600 nM T13852 CP45BX 11495124 EC50 = 6.5 nM T13852 CW51YT 11495139 IC50 = 5.7 nM T13852 CDE78J 11496072 EC50 = 0.12 nM T13852 CWL71C 11496105 EC50 = 1 nM T13852 CS5A1E 11501417 IC50 = 74 nM T13852 C7EOU1 11501764 IC50 = 5.1 nM T13852 CR1ME9 11501873 EC50 = 1.9 nM T13852 CS27OX 11502026 IC50 = 100 nM T13852 CRO87D 11503250 EC50 = 0.6 nM T13852 CDVR16 11503306 EC50 = 3 nM T13852 CL50IH 11503967 EC50 = 18.3 nM T13852 CC02BK 11510741 IC50 = 4.75 nM T13852 CS4LD8 11530826 EC50 = 1800 nM T13852 CK0Y6I 11531691 EC50 = 4.4 nM T13852 CQ6S5W 11531879 EC50 = 0.58 nM T13852 CAG0Y9 11540052 EC50 = 0.52 nM T13852 CTF1L4 11553135 EC50 = 282 nM T13852 CU0C3H 11553524 EC50 = 1.8 nM T13852 CR5ED7 11555202 IC50 = 0.84 nM T13852 CLP3O7 11567535 EC50 = 4.6 nM T13852 C52ZWY 11568129 EC50 = 0.8 nM T13852 C3BK8V 11568622 EC50 = 0.19 nM T13852 CVW6Q3 11575787 IC50 = 0.8 nM T13852 CB75ZP 11575913 EC50 < 0.08 nM T13852 C5NAQ2 11589375 EC50 = 2.6 nM T13852 C02XSU 11595314 EC50 = 520 nM T13852 C9F4YI 11597340 EC50 = 1.1 nM T13852 CXS54Q 11603220 IC50 = 4.5 nM T13852 C5BDY3 11603528 EC50 = 0.98 nM T13852 CCW90K 11603726 EC50 = 0.15 nM T13852 C96LNP 11604577 IC50 = 0.9 nM T13852 CKH3L4 11609496 EC50 = 30 nM T13852 CAN4Q9 11611053 EC50 = 0.9 nM T13852 C7I6ZU 11619303 EC50 = 0.072 nM T13852 C41XAE 11624780 EC50 = 3.4 nM T13852 CCY7J2 11626664 EC50 = 0.1 nM T13852 C4IMA6 11632823 EC50 = 0.93 nM T13852 CXZ8T6 11633613 EC50 = 6.3 nM T13852 C13VZP 11640578 EC50 = 1.9 nM T13852 CA8W5N 11646599 EC50 = 0.2 nM T13852 C21VTL 11647892 EC50 = 1.3 nM T13852 CYS5F1 11653967 IC50 = 2.2 nM T13852 C8TL6P 11654374 EC50 = 0.18 nM T13852 CMJ32O 11662328 EC50 = 0.3 nM T13852 CQTW52 11675496 EC50 = 5.1 nM T13852 C8CQ2N 11675907 EC50 = 4.7 nM T13852 CD4AO7 11676168 EC50 = 1.1 nM T13852 CCNU48 11678855 EC50 = 1 nM T13852 CR94XU 11682224 EC50 = 450 nM T13852 C3Q9JR 11682677 EC50 = 4 nM T13852 CVG41H 11682696 EC50 = 1.1 nM T13852 CQRA36 11683935 IC50 = 2.5 nM T13852 CCF80W 11689680 EC50 = 0.08 nM T13852 CTB2W7 11690483 EC50 = 1.4 nM T13852 C8XLO4 11690779 IC50 = 186 nM T13852 C0BR1U 11696807 IC50 = 8.2 nM T13852 CK5S1L 11697013 EC50 = 0.7 nM T13852 CL80RC 11697277 EC50 = 4.7 nM T13852 C2ZWP0 11697911 EC50 = 0.53 nM T13852 CK63OB 11705484 IC50 = 2000 nM T13852 C4G2OP 11743459 IC50 = 0.4 nM T13852 CZ6YN9 11752659 EC50 = 2.7 nM T13852 CJ98PB 11852048 EC50 = 21 nM T13852 CV3WI7 11852049 EC50 = 19 nM T13852 C2Z8AY 11852142 EC50 = 71 nM T13852 C3J8TH 11852143 EC50 = 2.6 nM T13852 C2FEG4 11852144 EC50 = 3.4 nM T13852 CRVF18 11852146 EC50 = 7 nM T13852 CLI76U 11852148 EC50 = 14 nM T13852 CEW5F3 11852233 EC50 = 1.2 nM T13852 C9D3UE 11852234 EC50 = 4.3 nM T13852 C0J2EH 11852237 EC50 = 1.1 nM T13852 C67GNU 11852437 EC50 = 0.4 nM T13852 CWF0P2 11852636 EC50 = 6.1 nM T13852 CI1S6O 11852848 EC50 = 1.7 nM T13852 CB67GQ 11852952 EC50 = 0.5 nM T13852 CH5W6S 11852953 EC50 = 1.2 nM T13852 CUBD18 11852955 EC50 = 1.5 nM T13852 C4N3DG 11853337 EC50 = 2.6 nM T13852 CMK7W8 11853338 EC50 = 10.7 nM T13852 CQ0V5W 11853576 EC50 = 5.1 nM T13852 C7YJM4 11853579 EC50 = 13.4 nM T13852 C09ZXI 11853580 EC50 = 1.1 nM T13852 CFUQ37 11853832 EC50 = 4.8 nM T13852 CU6M7E 11853834 EC50 = 1.5 nM T13852 CWR71V 11853835 EC50 = 2 nM T13852 CMJ71A 11853836 EC50 = 0.6 nM T13852 CKOR74 11854090 EC50 = 4.4 nM T13852 CQ78BJ 11854356 EC50 = 3.3 nM T13852 CS8E1K 11854607 EC50 = 1.2 nM T13852 CF7W9B 11854857 EC50 = 0.9 nM T13852 CLHA36 11869937 EC50 = 16 nM T13852 C1LMA8 11977818 EC50 = 1 nM T13852 CA9D8B 11977936 EC50 = 11 nM T13852 C03OUS 11977938 EC50 = 4 nM T13852 CUM5T9 11977939 EC50 = 5 nM T13852 CYE48W 11978048 EC50 = 4 nM T13852 CPSI96 11978050 EC50 = 8.5 nM T13852 CGS70F 11978162 EC50 = 6.5 nM T13852 COY96U 11978278 EC50 = 25 nM T13852 CDI32A 16038017 EC50 = 0.11 nM T13852 CE5OB2 16051482 EC50 = 117 nM T13852 C4TQR8 16105530 IC50 = 6640 nM T13852 CJ2E4B 16105541 IC50 = 4280 nM T13852 C65RDB 16188020 EC50 > 50000 nM T13852 CLA85D 16657820 EC50 = 0.5 nM T13852 CX71MV 16735046 EC50 = 454 nM T13852 CS0X4J 16736754 EC50 = 290 nM T13852 CG8J5U 16736755 EC50 = 158 nM T13852 CDK2Z5 16737130 EC50 = 520 nM T13852 CA9P2L 16737316 EC50 = 420 nM T13852 CZGM01 16737317 EC50 = 1600 nM T13852 C6FW1V 16737319 EC50 = 48 nM T13852 CC6W8M 16737345 EC50 = 620 nM T13852 CY7U2O 16737504 EC50 = 150 nM T13852 CR0B6Y 16737505 EC50 = 354 nM T13852 C58EWF 16737507 EC50 = 253 nM T13852 CU30WQ 16737509 EC50 = 424 nM T13852 CZ41LC 16737511 EC50 = 510 nM T13852 C4D2EF 16737513 EC50 = 2000 nM T13852 CU6Y0F 16737514 EC50 > 1000 nM T13852 CF4XN8 16737667 EC50 = 350 nM T13852 C6X5BR 16737668 EC50 = 440 nM T13852 C6M2FB 16737670 EC50 = 460 nM T13852 CDG57C 16737679 EC50 = 57 nM T13852 CIJF78 16737988 EC50 = 21 nM T13852 CRE74S 16738333 EC50 > 1000 nM T13852 CGAD08 17253208 EC50 = 33300 nM T13852 CIEK03 17253281 EC50 = 22250 nM T13852 CSQB62 17747461 EC50 = 1610 nM T13852 C6HB9A 21455530 IC50 = 7 nM T13852 CNV98Q 23121057 EC50 = 1500 nM T13852 C89BVX 23121067 EC50 = 280 nM T13852 CC75ZH 23121172 EC50 = 10 nM T13852 C0O5CY 23121189 EC50 = 1.7 nM T13852 CLZ45N 23121209 EC50 = 1300 nM T13852 C6DV2O 23121326 EC50 = 19 nM T13852 C7XK3S 23121338 EC50 = 57 nM T13852 CK6G0D 23121374 EC50 = 33 nM T13852 CI7RA6 23121393 EC50 = 20 nM T13852 C05RUE 23121412 EC50 = 1600 nM T13852 C6MJ4N 23121431 EC50 = 230 nM T13852 CF01WY 23121435 EC50 = 24 nM T13852 CME14G 23121436 EC50 = 36 nM T13852 C5AKM6 23121505 EC50 = 97 nM T13852 C14XBN 23121526 EC50 = 2700 nM T13852 CF1EU4 23121592 EC50 = 930 nM T13852 CYX03D 23121622 EC50 = 120 nM T13852 CUF57G 23729211 EC50 = 1.5 nM T13852 CEV1I3 23729229 EC50 = 1.5 nM T13852 C8R4SV 24744028 EC50 = 231 nM T13852 C2JGS9 24784418 EC50 = 0.7 nM T13852 C6I0ED 24812110 IC50 = 0.3 nM T13852 C0O9UG 24825338 EC50 = 0.08 nM T13852 CB82GW 24825339 EC50 = 0.44 nM T13852 CTH4S8 24850258 EC50 = 2890 nM T13852 C9QTZ3 24851764 EC50 = 5.7 nM T13852 CW2CD1 24851766 EC50 = 1.9 nM T13852 CUP73J 24863649 EC50 = 310 nM T13852 CJPA05 24863828 EC50 = 3030 nM T13852 CAP2X8 24863831 EC50 = 720 nM T13852 CU79ZI 24956673 EC50 = 47 nM T13852 C3RPZ4 24956674 EC50 = 67 nM T13852 CF9I1S 24956675 EC50 = 34 nM T13852 CYIJ40 24956676 EC50 = 112 nM T13852 CPT9J2 24957028 EC50 = 35 nM T13852 CU3R0D 24957029 EC50 = 19 nM T13852 CM7HQ5 24985395 EC50 = 7 nM T13852 CM2DL8 24985568 EC50 = 9 nM T13852 C8Z2JD 24985569 EC50 = 28 nM T13852 CEJ74C 24985745 EC50 = 4 nM T13852 CSXB36 24986380 EC50 = 0.01 nM T13852 C90SNU 24986381 EC50 = 2.512 nM T13852 C95TGD 24986921 EC50 = 12 nM T13852 C1TGE9 25008420 IC50 = 0.23 nM T13852 CV6EP4 25008421 EC50 = 700 nM T13852 C34RKU 25031771 EC50 = 0.3 nM T13852 CCJ17D 25032056 EC50 = 0.4 nM T13852 C8GUH0 25070493 EC50 = 7.9 nM T13852 C9WQC5 25072410 EC50 = 1.9 nM T13852 CCO54A 25074253 EC50 = 0.6 nM T13852 CLT95X 25110105 EC50 > 50000 nM T13852 CLW5E6 25110210 EC50 = 44900 nM T13852 CUZJ62 25110212 EC50 > 50000 nM T13852 C14EAK 25110484 EC50 = 859 nM T13852 C3S8QZ 25110485 EC50 = 6420 nM T13852 C01FRW 25110488 EC50 = 662 nM T13852 C07GXT 25110489 EC50 = 23100 nM T13852 CAP8T1 25110492 EC50 > 50000 nM T13852 CWUT04 25110494 EC50 > 50000 nM T13852 CXU68J 25110496 EC50 > 50000 nM T13852 CI2VH9 25110498 EC50 = 33100 nM T13852 CLEF36 25110499 EC50 = 4700 nM T13852 C8WAX0 25110500 EC50 > 50000 nM T13852 CS2WQ0 25110501 EC50 = 3260 nM T13852 CF50YO 25110510 EC50 > 50000 nM T13852 CJ3HS1 25110511 EC50 = 34150 nM T13852 CJ9CI6 25110521 EC50 > 25000 nM T13852 CP6A9Q 25110522 EC50 = 7600 nM T13852 C14CBE 25110524 EC50 > 25000 nM T13852 C1EM2P 25154344 EC50 = 3 nM T13852 C6RM3T 25182621 EC50 = 1160 nM T13852 C16VAH 25182623 EC50 = 16700 nM T13852 CGPM45 25182745 EC50 = 440 nM T13852 CFPX93 25182751 EC50 = 960 nM T13852 C68IMF 25182753 EC50 = 382 nM T13852 CQO8C7 25182755 EC50 = 1990 nM T13852 C1HT8Z 25182756 EC50 = 440 nM T13852 CM1T6P 25182757 EC50 = 2100 nM T13852 C5IV9U 25182758 EC50 = 700 nM T13852 CTK6S3 25182759 EC50 = 655 nM T13852 CX4G3V 25182761 EC50 = 973 nM T13852 C6X2BW 25182765 EC50 = 2710 nM T13852 CZQ4K9 25182766 EC50 = 65 nM T13852 CP1CA9 25182769 EC50 = 25 nM T13852 CGSU43 25182770 EC50 = 418 nM T13852 CF35EH 25182773 EC50 = 1.6 nM T13852 CS5DQ9 25182774 EC50 = 211 nM T13852 CU2JK0 25182778 EC50 = 73 nM T13852 CY16FK 25182780 EC50 > 20000 nM T13852 C0Y2ZH 25182781 EC50 = 1780 nM T13852 CM2NF8 25182782 EC50 = 2.9 nM T13852 CGEM35 25182899 EC50 = 12 nM T13852 CF6ZA0 25182902 EC50 = 39 nM T13852 CK9V3M 25182909 EC50 = 12 nM T13852 C4P1JM 25182910 EC50 = 7 nM T13852 CXF04D 25182915 EC50 = 12 nM T13852 CWOS48 25182921 EC50 = 104 nM T13852 CZ2WL8 25182923 EC50 = 35 nM T13852 C03BZW 25182925 EC50 = 94 nM T13852 CNYW93 25182926 EC50 = 19 nM T13852 C10HKX 25192001 EC50 = 0.077 nM T13852 CL7RV5 25192005 EC50 = 0.088 nM T13852 CB06TP 25192006 EC50 = 19.72 nM T13852 C2TO4H 25256388 EC50 = 6 nM T13852 CZ8Y9S 42610387 EC50 = 1.9 nM T13852 CHD3I5 42622931 EC50 = 0.6 nM T13852 C48TPJ 42630194 EC50 = 0.75 nM T13852 C9YBE0 42636433 EC50 = 7.943 nM T13852 CA81LQ 42636536 EC50 = 10 nM T13852 CS35FG 42636618 EC50 = 7.943 nM T13852 CNHI02 44124898 EC50 = 39.81 nM T13852 CDL1C8 44125170 EC50 = 5.012 nM T13852 CG5X4T 44125468 EC50 = 7.943 nM T13852 CNU5F1 44125469 EC50 = 316.23 nM T13852 CH3A1V 44125470 EC50 = 501.19 nM T13852 C51WHA 44125471 EC50 = 398.11 nM T13852 CRE0O1 44125588 EC50 = 5.012 nM T13852 CP1BF0 44125589 EC50 = 2.512 nM T13852 CS0H1B 44125704 EC50 = 39.81 nM T13852 C1YHG6 44128660 EC50 = 398.11 nM T13852 C4H5TR 44128662 EC50 = 125.89 nM T13852 CUQE25 44128745 EC50 = 1.995 nM T13852 CAH09Q 44128746 EC50 = 15.85 nM T13852 C31VJX 44128747 EC50 = 158.49 nM T13852 C7H4MR 44128748 EC50 = 2511.89 nM T13852 CH2ES5 44128819 EC50 = 630.96 nM T13852 CRIK86 44128821 EC50 = 316.23 nM T13852 CIL7J3 44128904 EC50 = 158.49 nM T13852 CY83JW 44128905 EC50 = 25.12 nM T13852 C19YHX 44128909 EC50 = 3.981 nM T13852 C47OXT 44128987 EC50 = 7.943 nM T13852 CW1DL9 44129063 EC50 = 79.43 nM T13852 CN5O1Y 44129065 EC50 = 39.81 nM T13852 CCTS05 44129140 EC50 = 25.12 nM T13852 CTV36P 44129142 EC50 = 125.89 nM T13852 CHL90M 44129143 EC50 = 50.12 nM T13852 C4EP2M 44129144 EC50 = 125.89 nM T13852 CP6MQ2 44129145 EC50 = 63.1 nM T13852 CABP65 44129218 EC50 = 79.43 nM T13852 C1BT4A 44129293 EC50 = 19.95 nM T13852 CAQ28H 44129298 EC50 = 19.95 nM T13852 CY1X3Z 44129373 EC50 = 5.012 nM T13852 CR9P3I 44136093 EC50 = 76 nM T13852 C0D3SH 44137116 EC50 = 157 nM T13852 CV08DP 44137120 EC50 = 4.6 nM T13852 C5WCA1 44137252 EC50 = 7.5 nM T13852 CG73ST 44138103 EC50 = 0.08 nM T13852 C0OY7M 44155199 EC50 = 2.9 nM T13852 C8ZCI1 44155200 EC50 = 0.59 nM T13852 C3OK4I 44156478 EC50 = 2.1 nM T13852 CQIL37 44156480 EC50 = 4.6 nM T13852 C9C3DA 44156481 EC50 = 0.61 nM T13852 CVUJ04 44199411 EC50 = 2.6 nM T13852 CNJ96W 44199424 EC50 = 0.5 nM T13852 C47CJM 44199450 EC50 = 2.1 nM T13852 CLR62S 44217168 EC50 = 14 nM T13852 CD3IM6 44217169 EC50 = 13 nM T13852 CC43PQ 44217170 EC50 = 7.1 nM T13852 C58BOP 44217502 EC50 = 1.1 nM T13852 C75XPC 44217654 EC50 = 2.8 nM T13852 CEHB49 44217839 EC50 = 1.3 nM T13852 CH0VO9 44217997 EC50 = 1.5 nM T13852 C7CB5P 44218002 EC50 = 0.2 nM T13852 C5L0QT 44218130 EC50 = 1.1 nM T13852 CO41AS 44218131 EC50 = 1.3 nM T13852 CI34VL 44218450 EC50 = 1 nM T13852 CWIC07 44218451 EC50 = 3.5 nM T13852 C7B1PL 44218479 EC50 = 1.2 nM T13852 C4F6RA 44218604 EC50 = 0.3 nM T13852 C25HOP 44218903 EC50 = 2.8 nM T13852 C4X5VS 44218906 EC50 = 5.1 nM T13852 CWNE68 44219368 EC50 = 8 nM T13852 C8AC7D 44219369 EC50 = 3.6 nM T13852 CKYJ71 44219370 EC50 = 4.1 nM T13852 CJ7M3E 44219525 EC50 = 2.1 nM T13852 CAY2S1 44219528 EC50 = 5.3 nM T13852 CH8CM7 44341291 IC50 = 17 nM T13852 CQR2G1 44341399 IC50 = 14 nM T13852 C95GIJ 44342175 Ki = 30 nM T13852 C7YT1J 44342219 EC50 = 260 nM T13852 C8NOT7 44342221 EC50 = 598.4 nM T13852 CCN68O 44342231 EC50 = 1805 nM T13852 CXJ08Y 44342244 EC50 = 397 nM T13852 C6LT8S 44342246 EC50 = 322.1 nM T13852 CLXY90 44342331 EC50 = 130 nM T13852 CI01UD 44342339 EC50 = 550 nM T13852 CAUQ90 44342468 EC50 = 82 nM T13852 CMKZ19 44344194 IC50 = 2.5 nM T13852 CLQ25X 44344210 IC50 = 30 nM T13852 C31BXA 44344270 IC50 = 0.5 nM T13852 CY7FC4 44344298 IC50 = 0.5 nM T13852 C1SP9M 44344338 IC50 = 360 nM T13852 C2D5LZ 44344360 IC50 = 12 nM T13852 CT4NW0 44344390 IC50 = 1.1 nM T13852 C9S2FH 44344404 IC50 = 6.6 nM T13852 CY9C1D 44344412 IC50 = 5.3 nM T13852 CLDU29 44344413 IC50 = 6.3 nM T13852 C91OKY 44344446 IC50 = 85 nM T13852 CL3CT8 44344456 IC50 = 15 nM T13852 CJ36UD 44394116 IC50 = 16 nM T13852 C5KA6D 44394117 IC50 = 1100 nM T13852 CU7L0K 44394153 IC50 = 49 nM T13852 CT8UN6 44394161 IC50 = 200 nM T13852 C9E6CF 44394169 IC50 = 89 nM T13852 C8H0XM 44394191 IC50 = 0.1 nM T13852 CH2A5S 44394211 IC50 = 220 nM T13852 CND39O 44394212 IC50 = 4.9 nM T13852 C84JPI 44394247 IC50 = 260 nM T13852 CA28OJ 44394273 IC50 = 0.16 nM T13852 CO0T1E 44394279 IC50 = 6.9 nM T13852 CE25XJ 44394289 EC50 = 1000 nM T13852 C0X4ZS 44394327 EC50 = 240 nM T13852 CL5BC6 44394330 IC50 = 260 nM T13852 CU3KA2 44394460 EC50 = 21 nM T13852 C24XDE 44394498 EC50 = 21 nM T13852 CZ14XU 44394521 EC50 = 330 nM T13852 CV9N2T 44394539 EC50 = 2900 nM T13852 C6XO8W 44394564 EC50 = 2100 nM T13852 CI75GS 44398012 EC50 = 9.8 nM T13852 CCFT02 44398049 EC50 = 150 nM T13852 CRYM50 44398058 EC50 = 7 nM T13852 CR3K9W 44398074 EC50 = 5100 nM T13852 C4DIT3 44398076 EC50 = 7.9 nM T13852 C3H2IY 44398170 EC50 = 6.4 nM T13852 CL5SY3 44398172 EC50 = 2700 nM T13852 CR4TH0 44406004 EC50 = 1 nM T13852 C3JF1Q 44406009 EC50 = 63.1 nM T13852 CK6J2H 44406749 EC50 = 19.95 nM T13852 CDY46P 44412165 IC50 = 1.2 nM T13852 CR2DT4 44412221 IC50 = 75 nM T13852 CRV34X 44412232 IC50 = 17 nM T13852 CV63YC 44412233 IC50 = 3.3 nM T13852 CQ1V3J 44412282 IC50 = 8 nM T13852 CB6KR7 44412294 IC50 = 4.5 nM T13852 CTV5M0 44412353 IC50 = 2 nM T13852 CN7K2O 44412364 IC50 = 0.8 nM T13852 CL1GJ3 44412415 IC50 = 5.7 nM T13852 CV28IK 44412416 IC50 = 0.7 nM T13852 CBM50W 44412428 IC50 = 2.7 nM T13852 C2US0I 44412578 EC50 = 1.6 nM T13852 CM46YR 44412604 EC50 = 290 nM T13852 C1LTZ6 44412605 EC50 = 1200 nM T13852 C28CAY 44412621 EC50 = 1.1 nM T13852 C9I7UV 44412622 EC50 > 10000 nM T13852 CNF3Y2 44412623 EC50 = 380 nM T13852 CG7T1N 44412643 EC50 > 10000 nM T13852 CF8J7Z 44412657 EC50 = 7.7 nM T13852 C05TUB 44412658 EC50 = 16 nM T13852 CH51GD 44412659 EC50 = 208 nM T13852 C93OLQ 44412660 EC50 > 10000 nM T13852 C0CA6R 44412661 EC50 = 14 nM T13852 C8J7HN 44412673 EC50 = 45 nM T13852 CL54DN 44412674 EC50 > 3600 nM T13852 C3M5SO 44412702 EC50 = 88 nM T13852 CGE62Q 44412703 EC50 = 38 nM T13852 C69HQV 44412704 EC50 = 0.23 nM T13852 CU23YP 44412720 EC50 = 360 nM T13852 CR75ED 44412721 EC50 = 94 nM T13852 C67MBH 44412755 IC50 = 0.6 nM T13852 C9G6HR 44412812 EC50 = 3.4 nM T13852 CX1C0G 44412813 EC50 = 0.2 nM T13852 C48CIX 44412814 EC50 = 570 nM T13852 CBUQ92 44412827 EC50 = 12 nM T13852 CT0UL5 44412828 EC50 = 0.16 nM T13852 C2AEO3 44412839 EC50 > 1000 nM T13852 CT4SG3 44412840 EC50 = 97 nM T13852 CB7X9U 44412841 EC50 = 2.8 nM T13852 CPHG35 44412853 EC50 = 19 nM T13852 CM8IK4 44412854 EC50 = 830 nM T13852 CUPK30 44412855 EC50 = 2.1 nM T13852 C34QEC 44412865 EC50 = 2.1 nM T13852 C4YAT1 44412866 EC50 = 1000 nM T13852 CBL87K 44412867 EC50 = 0.4 nM T13852 COA6Q1 44412868 EC50 = 3.2 nM T13852 C80JSN 44412882 EC50 = 0.5 nM T13852 C2WV6S 44412883 EC50 = 14 nM T13852 C84PLZ 44412908 EC50 = 2.4 nM T13852 C78DOK 44412936 EC50 = 0.07 nM T13852 CH6Z8V 44412962 EC50 = 467 nM T13852 C03WFR 44412970 EC50 = 9.5 nM T13852 C3MWD4 44412971 EC50 = 0.03 nM T13852 CR4DQ3 44412993 EC50 = 1.1 nM T13852 CJC06H 44412994 EC50 = 0.1 nM T13852 CH84GV 44413027 EC50 = 0.61 nM T13852 C2IMP5 44413039 EC50 = 0.28 nM T13852 C0CI2U 44413057 EC50 = 0.79 nM T13852 CT6EU7 44413274 IC50 = 25 nM T13852 CYO6R3 44413349 IC50 = 1.2 nM T13852 CH9NL4 44413365 IC50 = 2 nM T13852 CW8E0R 44413415 IC50 = 2.2 nM T13852 CYW5D3 44413430 IC50 = 7.9 nM T13852 CJ5S2H 44413446 IC50 = 1 nM T13852 CWRZ40 44413447 IC50 = 1.4 nM T13852 CVC61G 44413482 IC50 = 5.5 nM T13852 CWL92R 44422573 EC50 = 27 nM T13852 CW67ZB 44422578 EC50 = 33 nM T13852 C12CHR 44422579 EC50 = 30 nM T13852 C4MTP5 44422590 EC50 = 1200 nM T13852 C0I3LB 44422601 EC50 = 3.6 nM T13852 C2O7AP 44422604 EC50 = 2.1 nM T13852 C07YCS 44422605 EC50 = 68 nM T13852 C7O0PC 44422606 EC50 = 140 nM T13852 CTGM54 44437363 IC50 = 5500 nM T13852 CA9W0D 44437367 IC50 = 1300 nM T13852 CN8KQ2 44437369 IC50 = 4600 nM T13852 CLKG90 44437373 IC50 = 400 nM T13852 CD72FV 44437375 IC50 > 17000 nM T13852 C9P0DB 44437377 IC50 = 8900 nM T13852 CXLZ52 44437379 IC50 = 700 nM T13852 CP1HE8 44437382 IC50 = 400 nM T13852 CUT38N 44437384 IC50 = 190 nM T13852 C2WEQ7 44437392 IC50 = 1000 nM T13852 C5NF3R 44437395 IC50 = 520 nM T13852 CV2I8Q 44437397 IC50 > 2400 nM T13852 CS8MN3 44437400 IC50 = 370 nM T13852 CSM2Y0 44437403 IC50 > 8100 nM T13852 C5H8WL 44437406 IC50 = 1000 nM T13852 C61QXD 44437410 IC50 = 80 nM T13852 C6NIG7 44437412 IC50 > 20000 nM T13852 CREM62 44437415 IC50 = 340 nM T13852 CP1FN6 44437417 IC50 = 500 nM T13852 C0MNU1 44437420 IC50 = 98 nM T13852 C50PYC 44437422 IC50 = 130 nM T13852 C0W3FQ 44439850 EC50 = 0.21 nM T13852 CB4Z3I 44439851 EC50 = 0.31 nM T13852 C9SFT8 44439852 EC50 = 0.8 nM T13852 CS9H0L 44517795 EC50 = 1.2 nM T13852 CQF0I7 44547175 EC50 = 25.12 nM T13852 C0NMA9 44547315 EC50 = 0.01259 nM T13852 C5WQ8J 44547316 EC50 = 0.00631 nM T13852 CJNM95 44547318 EC50 = 0.2512 nM T13852 CX13MK 44547414 EC50 = 4.6 nM T13852 C2M5EO 44547415 EC50 = 10.3 nM T13852 C3TM9X 44547416 EC50 = 4 nM T13852 CZAM42 44547417 EC50 = 18 nM T13852 C4C0QA 44547418 EC50 = 6.3 nM T13852 CGZ84E 44547461 EC50 = 0.1995 nM T13852 C0Z5IV 44547555 EC50 = 68 nM T13852 CL8IZ9 44547556 EC50 = 11 nM T13852 CDQL02 44547557 EC50 = 11 nM T13852 C7DP3Z 44547558 EC50 = 18 nM T13852 CKU57J 44547560 EC50 = 1.63 nM T13852 CG6D3L 44547603 EC50 = 0.3981 nM T13852 CU3V6A 44547605 EC50 = 0.2512 nM T13852 CFI6C1 44547606 EC50 = 1.585 nM T13852 C5S0MH 44547608 EC50 = 100 nM T13852 C01LHF 44547705 EC50 = 45 nM T13852 CD4VY9 44547708 EC50 = 102 nM T13852 CB54DU 44547709 EC50 = 6.6 nM T13852 C4PI2K 44547710 EC50 = 6.1 nM T13852 C27WLJ 44547758 EC50 < 0.01 nM T13852 CRE1H3 44547861 EC50 = 1 nM T13852 CM46WV 44547862 EC50 = 5.3 nM T13852 CZKC47 44547863 EC50 = 1.5 nM T13852 CL2RF3 44547909 EC50 = 0.3162 nM T13852 CXMF34 44547910 EC50 = 199.53 nM T13852 C2OM1R 44547911 EC50 = 19.95 nM T13852 C3UR4T 44548010 EC50 = 2.7 nM T13852 CI1FJ7 44548011 EC50 = 38 nM T13852 CT4IE0 44548012 EC50 = 0.82 nM T13852 CH4F0V 44548058 EC50 = 39.81 nM T13852 C46GZY 44548059 EC50 = 0.3981 nM T13852 CF1JW9 44548061 EC50 = 0.05012 nM T13852 C2LWN0 44548170 EC50 = 1.3 nM T13852 CMYZ28 44548224 EC50 = 3.162 nM T13852 CV9GB5 44548226 EC50 = 1258.93 nM T13852 COU3R0 44565595 IC50 = 21 nM T13852 CP18DA 44565596 EC50 = 0.52 nM T13852 CO8AD3 44565597 EC50 = 2.9 nM T13852 C75UYT 44565621 IC50 = 30 nM T13852 CS13TE 44565622 IC50 = 1.2 nM T13852 CU1NS0 44565703 IC50 = 220 nM T13852 CIY08J 44565712 IC50 = 0.78 nM T13852 C16WTE 44565713 IC50 = 12 nM T13852 COH39N 44565714 EC50 = 1.1 nM T13852 CB1GT5 44565715 EC50 = 2.67 nM T13852 CAV3F9 44565716 EC50 = 2.2 nM T13852 C76DFZ 44565717 IC50 = 1.03 nM T13852 CMG7L1 44565738 EC50 = 7.3 nM T13852 CH8SJ9 44565739 EC50 = 10.2 nM T13852 CX9AZ4 44591249 EC50 = 2.4 nM T13852 C3NOY0 44591250 EC50 = 1.1 nM T13852 C3TAY6 44591264 EC50 = 2.1 nM T13852 CGCL62 44591265 EC50 = 0.55 nM T13852 C10TGI 44591266 EC50 = 0.45 nM T13852 C92QVU 44599024 EC50 = 119 nM T13852 CI3L4J 44599683 EC50 = 240 nM T13852 C0EI2G 44599686 EC50 = 42 nM T13852 CR1FP6 44599687 EC50 = 36 nM T13852 CRMO89 44600329 EC50 = 179 nM T13852 C1GW4T 44600476 EC50 = 2 nM T13852 C5I8AH 44600484 EC50 = 62 nM T13852 CPM41D 44600642 EC50 = 26 nM T13852 CS3RZ6 44600643 EC50 = 33 nM T13852 CJR1B7 44600645 EC50 = 38 nM T13852 CB94AO 44601271 EC50 = 5880 nM T13852 C7QH2J 44602504 EC50 = 0.073 nM T13852 C91ESJ 44623997 EC50 = 0.077 nM T13852 C36BGS 44623999 EC50 = 16 nM T13852 C78ATE 44624002 EC50 = 1.7 nM T13852 C6SBV7 44624067 EC50 = 0.09 nM T13852 CI04UZ 44624068 EC50 = 26 nM T13852 CQ7CL5 44624071 EC50 = 0.44 nM T13852 CAGN32 44624139 EC50 = 55.8 nM T13852 CA0W3D 44624140 EC50 = 159 nM T13852 CIOD72 44624141 EC50 = 0.087 nM T13852 CI6Z3Q 44624142 EC50 = 0.49 nM T13852 C20RVZ 44624203 EC50 = 0.45 nM T13852 CXLS19 44624204 EC50 = 3.68 nM T13852 CS5K3Q 44624207 EC50 = 141 nM T13852 C8PS4D 44624270 EC50 = 4.58 nM T13852 C7MJV8 44625666 EC50 = 18 nM T13852 CX2T3Z 44625749 EC50 = 11 nM T13852 CK69AU 44625750 EC50 = 94 nM T13852 CKS69U 44625752 EC50 = 0.4 nM T13852 CV5GL3 44625753 EC50 = 1.4 nM T13852 CZUT65 45376040 EC50 = 1.6 nM T13852 C7JFL9 45376041 EC50 = 2.17 nM T13852 CDV7R4 45376042 EC50 = 371 nM T13852 CT0K1S 45376237 IC50 = 500 nM T13852 C9A0ST 45376238 IC50 > 10000 nM T13852 CQK87P 45376239 IC50 = 326 nM T13852 CD7KF0 45376240 IC50 = 702 nM T13852 C5P2TE 45376573 EC50 > 10000 nM T13852 CYOW10 45377016 IC50 = 4.8 nM T13852 C7D3LB 45377018 IC50 = 26 nM T13852 C5N1YS 45377019 IC50 = 14 nM T13852 CN0A4O 45377161 IC50 = 2800 nM T13852 CR32YA 45377248 EC50 = 1 nM T13852 CSVU96 45377524 EC50 = 4000 nM T13852 C25PTU 45377580 IC50 = 48 nM T13852 C6T4QB 45377662 EC50 = 0.3 nM T13852 C85SQO 45377797 EC50 = 2.4 nM T13852 CWQY86 45377937 EC50 = 9 nM T13852 C9AZ0K 45377938 EC50 = 3 nM T13852 CB9O1N 45377940 EC50 = 47 nM T13852 C8ELI4 45378010 IC50 = 6.8 nM T13852 CH0Z5C 45378095 EC50 = 44 nM T13852 C5P7LK 45378098 EC50 = 4.7 nM T13852 C73DCB 46174905 EC50 = 0.041 nM T13852 CPU02J 46190696 IC50 = 13 nM T13852 CVDK53 46204808 EC50 = 0.64 nM T13852 C5MX8L 46204811 EC50 = 0.81 nM T13852 C78PDO 46205128 EC50 = 0.62 nM T13852 C1GEB0 46205132 EC50 = 1.2 nM T13852 C96WMQ 46205452 EC50 = 3.1 nM T13852 C1YQM5 46205453 EC50 = 21 nM T13852 C1RV6W 46205455 EC50 = 4.7 nM T13852 CV1G4W 46205774 EC50 = 1.6 nM T13852 CLI75U 46205775 EC50 = 1.1 nM T13852 CDA30X 46206103 EC50 = 0.84 nM T13852 COR39P 46206105 EC50 = 3.6 nM T13852 CHOV03 46206106 EC50 = 3 nM T13852 CQKV71 46206107 EC50 = 2 nM T13852 C1THR5 46206435 EC50 = 4.2 nM T13852 CSTA18 46224712 EC50 = 25 nM T13852 C4QB8F 46224713 EC50 = 16 nM T13852 C4HN6L 46224714 EC50 = 26 nM T13852 CF75RO 46224715 EC50 = 11 nM T13852 C6R9SJ 46224716 EC50 = 119 nM T13852 CB56OX 46224767 EC50 = 7 nM T13852 CHC1D9 46224768 EC50 = 17 nM T13852 C15WRO 46224769 EC50 = 2 nM T13852 CMW59H 46225233 EC50 > 10000 nM T13852 CV5T1F 46225282 EC50 > 10000 nM T13852 CF74HE 46225283 EC50 > 10000 nM T13852 C6XAU7 46225284 EC50 = 280 nM T13852 CL4H8B 46225285 EC50 > 10000 nM T13852 CQ6WU0 46236268 EC50 = 102 nM T13852 CUE6F1 46236269 EC50 = 147 nM T13852 C4NDW1 46236270 EC50 = 103 nM T13852 C01WTY 46236271 EC50 = 202 nM T13852 CV8LH3 46236272 EC50 = 347 nM T13852 CY75PB 46236273 EC50 = 584 nM T13852 CN8IP7 46236274 EC50 = 58 nM T13852 CEAU68 46236398 EC50 = 282 nM T13852 CI5C6D 46236399 EC50 = 10 nM T13852 CDP2R8 46236400 EC50 = 479 nM T13852 C7OUC4 46236401 EC50 > 10000 nM T13852 CW3H8J 46236402 EC50 = 55 nM T13852 C7I3DZ 46236403 EC50 = 110 nM T13852 COV15E 46236404 EC50 = 78 nM T13852 C5XR6Q 46236517 EC50 = 154 nM T13852 CUN5S8 46236518 EC50 = 72 nM T13852 CZAQ79 46236519 EC50 = 179 nM T13852 CB2PV6 46236520 EC50 = 124 nM T13852 CO2YA0 46236521 EC50 = 54 nM T13852 C9SNG5 46236522 EC50 = 31 nM T13852 CZU24S 46236523 EC50 = 47 nM T13852 CKZ0M4 46236660 EC50 = 106 nM T13852 CJOW38 46236661 EC50 = 259 nM T13852 C3O7UR 46236662 EC50 = 251 nM T13852 C8MO1E 46236663 EC50 = 875 nM T13852 C9YXI2 46236664 EC50 = 356 nM T13852 CQ6K2M 46236665 EC50 = 630 nM T13852 CI69FH 46236666 EC50 = 925 nM T13852 CN2O7F 46236805 EC50 = 1815 nM T13852 CG8BV2 46236806 EC50 = 1237 nM T13852 C8IF1Z 46236807 EC50 = 122 nM T13852 C46YWF 46236808 EC50 = 225 nM T13852 CWE42H 46236809 EC50 = 37 nM T13852 C8GOC2 46236810 EC50 = 200 nM T13852 CU2F3J 46236811 EC50 = 201 nM T13852 CP0J7W 46236929 EC50 = 224 nM T13852 CDLX95 46236930 EC50 = 148 nM T13852 C43CIM 46236931 EC50 = 1038 nM T13852 CG4O8A 46236932 EC50 = 185 nM T13852 CST73W 46236933 EC50 = 752 nM T13852 CP52YF 46236934 EC50 = 444 nM T13852 C1L6YP 46236935 EC50 > 10000 nM T13852 C1SC0X 46237046 EC50 = 6452 nM T13852 CA7W1B 46237047 EC50 > 10000 nM T13852 CJGE86 46237048 EC50 > 10000 nM T13852 CM3B0H 46237049 EC50 = 408 nM T13852 C23JZF 46237050 EC50 = 102 nM T13852 CV4HT8 46237051 EC50 = 98 nM T13852 CL4R3O 46237052 EC50 = 58 nM T13852 C2RJF5 46237175 EC50 = 143 nM T13852 CSW4X8 46237176 EC50 = 8631 nM T13852 CZKV91 46237177 EC50 = 1414 nM T13852 C21EUB 46237178 EC50 = 343 nM T13852 CPT48C 46237179 EC50 = 11 nM T13852 CZ01WY 46237180 EC50 = 12 nM T13852 C3PVA2 46237828 EC50 = 200 nM T13852 C0J8CN 46238363 EC50 = 62 nM T13852 C8N6IR 46238364 EC50 > 10000 nM T13852 C7Q8XW 46238365 EC50 = 990 nM T13852 C0Q7IH 46238366 EC50 = 186 nM T13852 C2M9XO 46835914 EC50 = 0.71 nM T13852 C9CR0E 46835922 EC50 = 0.27 nM T13852 C2XO4K 46846820 EC50 = 0.98 nM T13852 CFH04W 46846899 EC50 = 0.27 nM T13852 CIO26E 46846900 EC50 = 0.56 nM T13852 CF41CL 46846901 EC50 = 1.6 nM T13852 C6DKO5 46846902 EC50 = 5.3 nM T13852 C80DQI 46846904 EC50 = 0.54 nM T13852 CEF91N 46846906 EC50 = 0.44 nM T13852 CA2W3P 46846912 EC50 = 0.99 nM T13852 CQ1N4Z 46846913 EC50 = 0.3 nM T13852 CG3RT7 46846915 EC50 = 0.39 nM T13852 CSU08A 46846921 EC50 = 3.2 nM T13852 CH8TL1 46847145 EC50 = 0.82 nM T13852 CI63SP 46847146 EC50 = 1 nM T13852 CC5JQ3 46847147 EC50 = 3.4 nM T13852 CTKC40 46847148 EC50 = 0.21 nM T13852 CQY5P8 46866185 EC50 = 19 nM T13852 C6LJ7A 46866186 EC50 = 44 nM T13852 CD2HV5 46872048 IC50 = 120 nM T13852 CP0A4M 46872507 IC50 > 10000 nM T13852 C13OBR 46872619 IC50 = 166 nM T13852 CB8IG2 46872620 IC50 = 217 nM T13852 CL69YZ 46872622 IC50 = 4230 nM T13852 CTM7O9 46872625 IC50 > 10000 nM T13852 CLS29B 46872626 IC50 = 362 nM T13852 C87CZT 46880278 EC50 = 12100 nM T13852 CA12XO 46880279 EC50 = 7300 nM T13852 C0W7IX 46880280 EC50 = 9 nM T13852 C1V3MY 46880712 EC50 > 20000 nM T13852 CH94GB 46880713 EC50 > 20000 nM T13852 C6MD9C 46880760 EC50 > 20000 nM T13852 CAD23F 46880801 EC50 = 375 nM T13852 CZ15OM 46880838 EC50 > 20000 nM T13852 C9OWJ3 46880839 EC50 > 20000 nM T13852 CZ54HF 46880876 EC50 > 20000 nM T13852 C2WU1C 46880877 EC50 > 20000 nM T13852 COGW78 46880925 EC50 = 193 nM T13852 C0FX1T 46880964 EC50 = 6 nM T13852 C50RIA 46881536 EC50 = 208 nM T13852 CVZ0F8 46881537 EC50 = 33 nM T13852 CH12FR 46881538 EC50 = 20 nM T13852 CU2I6S 46881580 EC50 = 238 nM T13852 CQZ59G 46881623 EC50 = 3 nM T13852 CW6RX2 46881847 EC50 = 0.85 nM T13852 CE32QB 46881848 EC50 = 110 nM T13852 CAHC81 46881875 EC50 = 20 nM T13852 C0BOR7 46881876 EC50 = 240 nM T13852 CCS12Z 46881877 EC50 = 960 nM T13852 C3QMS1 46881912 EC50 = 460 nM T13852 CY3S0L 46883880 EC50 = 13.65 nM T13852 CTL89X 46884020 EC50 = 0.018 nM T13852 CYJL86 46885693 IC50 = 21 nM T13852 C17RPW 46885694 IC50 > 10000 nM T13852 C7SB8P 46885695 IC50 = 150 nM T13852 C1I9TX 46885696 IC50 = 500 nM T13852 CC60OX 46885742 IC50 = 3.4 nM T13852 CEQ7V1 46885743 IC50 = 0.8 nM T13852 CF5V3E 46885744 IC50 = 1.3 nM T13852 COL9E8 46885745 IC50 = 6 nM T13852 CJ21TY 46885796 EC50 = 1.44 nM T13852 CGTR17 46885797 IC50 = 6.4 nM T13852 CZDL71 46885798 EC50 = 22.4 nM T13852 CL0C6G 46885873 EC50 = 1.1 nM T13852 CWV3O6 46886019 EC50 = 1.8 nM T13852 CV71KJ 46928129 EC50 = 100 nM T13852 CV6WT1 46929213 EC50 = 32 nM T13852 CG9X7Z 49830722 IC50 = 333 nM T13852 CS6JN0 49830723 IC50 = 680 nM T13852 CJ3CQ5 49830724 IC50 = 256 nM T13852 CS1NI2 49830725 IC50 = 1060 nM T13852 C84YOW 49830828 IC50 = 835 nM T13852 C3SAE6 49830919 IC50 = 221 nM T13852 CS25XW 49835989 EC50 = 68 nM T13852 C5Z6RM 49839234 EC50 = 0.03 nM T13852 CL64TH 49842175 EC50 = 1.259 nM T13852 CPJ25K 49847296 EC50 = 100 nM T13852 C8KQB9 49848139 EC50 = 0.1995 nM T13852 CNA18Z 49848426 EC50 = 63.1 nM T13852 CU86ZT 49848427 EC50 = 3.162 nM T13852 CAL07G 49848428 EC50 = 630.96 nM T13852 CJGR71 49848429 EC50 = 5.012 nM T13852 C29KYX 49848430 EC50 = 3.981 nM T13852 C4BXP1 49848557 EC50 = 1.585 nM T13852 CZG98A 49848559 EC50 = 125.89 nM T13852 CKD3E5 49848560 EC50 = 5.012 nM T13852 CK29IW 49848561 EC50 = 6.31 nM T13852 CHLR06 49848655 EC50 = 3.162 nM T13852 CQ32CR 49848656 EC50 = 1.259 nM T13852 CJM64G 49848776 EC50 = 1.259 nM T13852 CM6ZD1 49848777 EC50 = 3.981 nM T13852 C07NGT 49848778 EC50 = 2.512 nM T13852 C74KWB 49848898 EC50 = 3.162 nM T13852 CMV6Y2 49868651 EC50 = 1.2 nM T13852 CA7M0E 49871977 EC50 = 0.4 nM T13852 CE7I5G 49872065 EC50 = 0.6 nM T13852 C6QH3P 49872066 EC50 = 7.3 nM T13852 CHJ97Z 49872506 EC50 = 0.04 nM T13852 CW3L7B 49872507 EC50 = 220 nM T13852 CK92OQ 49872598 EC50 = 150 nM T13852 CBN81A 49872599 EC50 = 0.41 nM T13852 C48GBV 49872600 EC50 = 0.04 nM T13852 CVR6A3 49872602 EC50 = 0.3 nM T13852 CSI84V 49872695 EC50 = 19 nM T13852 C7LC8S 49872696 EC50 = 10000 nM T13852 C9T4VC 49872697 EC50 = 400 nM T13852 C4Q8MN 49872698 EC50 = 10000 nM T13852 C08IFS 49872790 EC50 = 290 nM T13852 CJ16ZQ 49872791 EC50 = 1.2 nM T13852 CEP4M8 49872977 EC50 = 1.7 nM T13852 C7NTH3 49872979 EC50 = 0.14 nM T13852 CY3XQ1 49872980 EC50 = 0.04 nM T13852 C7WH3E 49872981 EC50 = 0.67 nM T13852 C36WZL 49872982 EC50 = 2.1 nM T13852 C7GD8K 49873101 EC50 = 0.04 nM T13852 CWH13K 49873102 EC50 = 0.04 nM T13852 C5R2FI 49873105 EC50 = 11 nM T13852 C6GI5F 49873106 EC50 = 0.48 nM T13852 CV1L7N 49873196 EC50 = 6.8 nM T13852 CZ5AI3 49873197 EC50 = 1.7 nM T13852 C9PGJ0 49873283 EC50 = 0.15 nM T13852 C7LQ8B 50923120 EC50 = 30 nM T13852 CT56SE 50923123 EC50 = 22 nM T13852 CDG10V 50923126 EC50 = 2.3 nM T13852 CH10BV 50923273 IC50 = 7 nM T13852 CFQV13 50923275 EC50 = 6.9 nM T13852 C69IWK 50923276 IC50 = 25 nM T13852 CD75CR 50923423 IC50 = 9.4 nM T13852 CU62PH 50923424 EC50 = 11 nM T13852 C8X0ZH 50923425 IC50 = 13 nM T13852 CC2VU3 50923427 IC50 = 5.8 nM T13852 C5HA0M 50925181 IC50 = 0.69 nM T13852 CBL82V 50925335 IC50 = 4 nM T13852 CNM61U 50925336 IC50 = 0.21 nM T13852 CH0B8K 50925337 EC50 = 3.5 nM T13852 CY15ZW 51036168 EC50 = 0.5 nM T13852 CVDN46 51346809 EC50 = 21 nM T13852 C2W8LE 51346934 EC50 = 42 nM T13852 C48OFS 53317713 EC50 = 94 nM T13852 CFL29U 53318124 EC50 = 41 nM T13852 C6QY0V 53318125 EC50 = 138 nM T13852 CG1KZ7 53318790 EC50 = 741 nM T13852 CI1D3M 53319457 EC50 = 144 nM T13852 C45YTZ 53319458 EC50 = 35 nM T13852 CER0W1 53320088 EC50 = 13 nM T13852 CU2P1O 53320107 EC50 = 49 nM T13852 C9SVK4 53320108 EC50 = 159 nM T13852 C17BHO 53320170 EC50 = 1500 nM T13852 CWU0X3 53320363 EC50 = 42 nM T13852 CF3VN5 53322061 EC50 = 199 nM T13852 C5H4NQ 53322110 EC50 = 520 nM T13852 C56HPB 53322715 EC50 = 325 nM T13852 CA1W8U 53322735 EC50 = 21 nM T13852 CJQ3A1 53322736 EC50 = 126 nM T13852 CI06MU 53322737 EC50 = 26 nM T13852 CL14WS 53322738 EC50 = 77 nM T13852 CG17KO 53323419 EC50 = 1600 nM T13852 C1FXC6 53323420 EC50 = 38 nM T13852 CL4OZ7 53323421 EC50 = 33 nM T13852 CEP7Z4 53324301 EC50 = 1810 nM T13852 C5TCI2 53324339 EC50 = 42 nM T13852 CA87QM 53324746 EC50 = 221 nM T13852 CLHX41 53325368 EC50 > 6250 nM T13852 C7X8YO 53325380 EC50 = 54 nM T13852 CRA75F 53326036 EC50 = 429 nM T13852 C7MR1A 53326037 EC50 = 3980 nM T13852 C9T4QX 53326615 EC50 = 6720 nM T13852 CVD5A8 53326641 EC50 = 33 nM T13852 CQDP84 53326886 EC50 = 30 nM T13852 C1DYT0 53358422 IC50 = 6400 nM T13852 CC7DZ4 53362086 EC50 = 0.021 nM T13852 C9CT8N 53373573 EC50 = 1 nM T13852 CG3FA9 53492750 EC50 = 3.162 nM T13852 CW69RX 54576288 EC50 = 0.1 nM T13852 C78NBU 54576289 EC50 = 0.2512 nM T13852 CU2Q1F 54576290 EC50 = 0.2512 nM T13852 CVA4I0 54576291 EC50 = 0.1585 nM T13852 C1BQ9K 54576499 EC50 = 3.981 nM T13852 C4P8DY 54576501 EC50 = 7.943 nM T13852 CSAV94 54576503 EC50 = 0.7943 nM T13852 CTUN47 54576721 EC50 = 0.7943 nM T13852 C61UKW 54579593 EC50 = 15.85 nM T13852 C5M2PI 54580603 IC50 > 20000 nM T13852 CWNO65 54582607 IC50 = 5300 nM T13852 CI20JA 54756906 EC50 = 19.95 nM T13852 CCG08B 54756907 EC50 = 19.95 nM T13852 CK50BF 54756908 EC50 = 7.943 nM T13852 CILG27 54758399 EC50 = 19.95 nM T13852 CU62DN 54764919 EC50 = 35 nM T13852 CHLD32 56834955 EC50 = 20 nM T13852 CA80UC 56835064 EC50 = 0.55 nM T13852 CKRB95 56835157 EC50 = 2840 nM T13852 CDN71L 56835182 EC50 = 17 nM T13852 CR9TC2 56948654 IC50 = 13 nM T13852 C7HYC3 56948659 EC50 = 130 nM T13852 C64ORS 56951563 EC50 = 18 nM T13852 C5GW1D 56953916 IC50 > 1000 nM T13852 CGSK38 56953917 IC50 = 33 nM T13852 C6A2WB 56953918 IC50 = 211 nM T13852 C0JZW3 56953919 IC50 = 96 nM T13852 CQIV20 56953920 IC50 > 10000 nM T13852 CBIH06 56954024 IC50 = 13 nM T13852 CB4GY3 56954025 IC50 = 152 nM T13852 CO5HX9 56954026 IC50 > 10000 nM T13852 CX6Z1Q 56954027 IC50 = 743 nM T13852 CHJV61 56954145 IC50 > 10000 nM T13852 CJIZ72 56954146 IC50 = 752 nM T13852 C85JVD 56954147 IC50 = 181 nM T13852 CNUC26 56954148 IC50 = 8281 nM T13852 CHY98A 56954159 IC50 > 1000 nM T13852 CY6H7G 56954240 IC50 = 239 nM T13852 CD32ZL 56954241 IC50 = 84 nM T13852 CGRC25 56954242 IC50 = 84.7 nM T13852 CRT0Y2 56954243 IC50 = 158 nM T13852 CBE76J 56954244 IC50 = 492 nM T13852 CF2Q9V 56955980 EC50 > 50000 nM T13852 C0I9ED 56955982 EC50 > 50000 nM T13852 C1LAY2 57335019 EC50 = 0.2 nM T13852 CW9QP5 57390104 EC50 = 570 nM T13852 CM36YP 57390142 EC50 = 1300 nM T13852 CN6LF0 57390143 EC50 > 20000 nM T13852 C8A1WC 57390144 EC50 = 2710 nM T13852 C1RK0O 57390238 EC50 = 3010 nM T13852 CKWG20 57390239 EC50 = 720 nM T13852 C5PX7M 57390794 EC50 = 2410 nM T13852 CW6VG3 57390795 EC50 = 2 nM T13852 CJSY48 57391111 EC50 = 372 nM T13852 CFP30K 57391212 EC50 > 100 nM T13852 CB2O0K 57391213 EC50 = 297 nM T13852 C4EF3Z 57391457 EC50 = 110 nM T13852 C3O4YQ 57391821 EC50 = 20 nM T13852 CT27YQ 57391849 EC50 = 3 nM T13852 CV7ZY6 57391886 EC50 = 2370 nM T13852 CHMJ97 57391887 EC50 = 1960 nM T13852 CK3X6Y 57391920 EC50 = 70 nM T13852 CO0CG8 57391921 EC50 = 41 nM T13852 C1HQ3L 57392027 EC50 = 4470 nM T13852 C2QK1U 57392608 EC50 = 8 nM T13852 CE0K1G 57392609 EC50 = 196 nM T13852 CWSR47 57392652 EC50 = 3 nM T13852 CDNC42 57392979 EC50 = 7.2 nM T13852 CAV7Y3 57393474 EC50 = 1100 nM T13852 C9B2VK 57393585 EC50 = 4.5 nM T13852 CO7A0R 57393586 EC50 = 5 nM T13852 C0MAT8 57393649 EC50 = 42 nM T13852 CZT94U 57394329 EC50 = 19 nM T13852 COJI42 57394406 EC50 = 2820 nM T13852 C5OES7 57394720 EC50 = 369 nM T13852 C58VEZ 57394721 EC50 = 1.2 nM T13852 C4F0IJ 57394951 EC50 = 35 nM T13852 CU0Z7A 57394952 EC50 = 21 nM T13852 C5WPX0 57395262 EC50 = 2.7 nM T13852 CLM47H 57395264 EC50 = 0.85 nM T13852 CB5SI2 57395297 EC50 = 30 nM T13852 CD1H8X 57395369 EC50 = 430 nM T13852 CR16YK 57395370 EC50 = 4100 nM T13852 CSG64Z 57395371 EC50 = 29 nM T13852 CGTY01 57395372 EC50 = 190 nM T13852 CP56XE 57395373 EC50 = 1100 nM T13852 CZS2J6 57395374 EC50 = 2900 nM T13852 CM74JH 57395471 EC50 = 816 nM T13852 CY5H6S 57396084 EC50 = 0.5 nM T13852 CFR73W 57396172 EC50 = 3 nM T13852 C91AGD 57396479 EC50 = 4.9 nM T13852 C74BYV 57396486 EC50 = 1.1 nM T13852 CN98GO 57396699 EC50 = 8.5 nM T13852 C8EUA6 57397066 EC50 = 75 nM T13852 C9MDA7 57397196 EC50 = 49 nM T13852 CPY57D 57397320 EC50 = 250 nM T13852 C3KS0A 57397321 EC50 = 18 nM T13852 C9HB5I 57397896 EC50 = 478 nM T13852 C57RHP 57397897 EC50 = 2 nM T13852 C3Q8JD 57397984 EC50 = 45 nM T13852 C8SB0Y 57398267 EC50 = 9.8 nM T13852 C8GNR7 57398268 EC50 = 75 nM T13852 C6NIS0 57398468 EC50 = 6.5 nM T13852 C4RPA5 57398469 EC50 = 850 nM T13852 CR39MB 57398470 EC50 > 20000 nM T13852 CE90LI 57398471 EC50 = 600 nM T13852 CUPB85 57398603 EC50 = 9 nM T13852 CG2F3T 57398732 EC50 = 3630 nM T13852 CJ8LF5 57398802 EC50 = 3 nM T13852 CD2H4N 57398845 EC50 = 6.5 nM T13852 CH2C9P 57398870 EC50 = 680 nM T13852 CZPO40 57398897 EC50 = 210 nM T13852 CT7E0J 57398996 EC50 = 1800 nM T13852 CXO9I1 57398998 EC50 = 287 nM T13852 CY98KJ 57399545 EC50 = 15 nM T13852 CLH87C 57399546 EC50 = 0.6 nM T13852 CJVQ54 57399579 EC50 = 2 nM T13852 CWBS53 57399928 EC50 = 4.3 nM T13852 C1Y9JG 57399929 EC50 = 41 nM T13852 C3HWU8 57400134 EC50 = 30 nM T13852 CX2R7O 57400135 EC50 = 60 nM T13852 C0EH7G 57400136 EC50 = 34 nM T13852 CVDZ56 57400137 EC50 = 200 nM T13852 C4A5EH 57400476 EC50 = 0.6 nM T13852 CPB4E0 57400520 EC50 = 14 nM T13852 C93FBE 57400521 EC50 = 7.5 nM T13852 CBE5U1 57400584 EC50 = 1170 nM T13852 CFS52K 57400585 EC50 = 42 nM T13852 CLGZ16 57400586 EC50 = 310 nM T13852 CXC10U 57400587 EC50 = 450 nM T13852 CQRU15 57400588 EC50 = 200 nM T13852 CS3I9U 57400714 EC50 = 34 nM T13852 CM8S5O 57401335 EC50 = 0.3 nM T13852 C08KNY 57401336 EC50 = 0.5 nM T13852 C3EWZ1 57401701 EC50 = 4.2 nM T13852 CXCY47 57401702 EC50 = 406 nM T13852 C5SC8F 57402192 EC50 = 2720 nM T13852 C57BKF 57402280 EC50 = 0.66 nM T13852 C5PVG3 57402282 EC50 = 0.37 nM T13852 C39PIE 57402284 EC50 = 1.1 nM T13852 CBP4S0 57402328 EC50 = 13 nM T13852 C86CHT 57402358 EC50 = 100 nM T13852 C5C7JK 57402390 EC50 = 2720 nM T13852 CHO08Y 57402391 EC50 = 24 nM T13852 CUZB73 57402392 EC50 = 60 nM T13852 CEH9D3 57403052 EC50 = 123 nM T13852 CI6J3E 57403053 EC50 = 3 nM T13852 CZM50H 57403429 EC50 = 1 nM T13852 CG2L6N 57403430 EC50 = 24 nM T13852 C3XV6B 57403435 EC50 = 37 nM T13852 CA39YG 57403436 EC50 = 54 nM T13852 CUN62P 57403950 EC50 > 100000 nM T13852 C6S0XI 57404009 EC50 = 4 nM T13852 CGE71H 57404012 EC50 = 4.5 nM T13852 CR7AU1 57404343 EC50 = 12.59 nM T13852 CO8JI5 57404344 EC50 = 1.259 nM T13852 CT9UR5 57404356 EC50 = 6.31 nM T13852 C0F5NL 57437353 EC50 = 0.6 nM T13852 CN49YH 57437389 EC50 = 1.3 nM T13852 C1QY9C 57505797 EC50 = 7.943 nM T13852 CDH87C 57505996 EC50 = 3.981 nM T13852 C3T2KX 57508868 EC50 = 1.6 nM T13852 CLF0Q9 57522810 EC50 = 10 nM T13852 C6X2YS 57522811 EC50 = 100 nM T13852 C52LBR 57522812 EC50 = 0.2512 nM T13852 CN0JL5 57522815 EC50 = 0.01585 nM T13852 CAZ1C6 57522939 EC50 = 0.01995 nM T13852 C6K0OG 57522940 EC50 = 199.53 nM T13852 CVS1Y9 57522941 EC50 = 1584.89 nM T13852 C0A1JE 57554662 IC50 > 30000 nM T13852 CLG2V4 57554674 IC50 < 1 nM T13852 CE5CS7 57570456 EC50 = 1500 nM T13852 C3UX5B 57570459 EC50 = 0.6 nM T13852 C7V4JG 57570461 EC50 = 2.6 nM T13852 CBF40Z 57570463 EC50 = 0.6 nM T13852 CGA79V 57570467 EC50 = 17 nM T13852 CY2N7Z 57570471 EC50 = 10000 nM T13852 CYW65N 57570476 EC50 = 1.6 nM T13852 C15XEN 57570479 EC50 = 61 nM T13852 C1KQE3 57570480 EC50 = 10000 nM T13852 CWMO74 57570481 EC50 = 120 nM T13852 CYB43R 57570486 EC50 = 0.4 nM T13852 C3AD7V 57570487 EC50 = 15 nM T13852 C0XE8J 57570490 EC50 = 640 nM T13852 CTZ20W 57570492 EC50 = 300 nM T13852 CJLX28 57570497 EC50 = 2 nM T13852 CA9CY8 57570498 EC50 = 0.3 nM T13852 C14RIK 57570499 EC50 = 9 nM T13852 C3U6YI 57570502 EC50 = 16 nM T13852 CZ19YS 57570503 EC50 = 2.2 nM T13852 CVIQ79 57570504 EC50 = 8 nM T13852 COE91B 57699087 Ki = 249 nM T13852 CH78XN 58329579 EC50 = 22 nM T13852 C4CM5G 58329587 EC50 = 1.1 nM T13852 CS87YX 58329594 EC50 = 150 nM T13852 C8ZW9H 58329596 EC50 = 38 nM T13852 CKHA51 58329600 EC50 = 2.3 nM T13852 CPJ03Q 58329604 EC50 = 0.49 nM T13852 CO95GF 58329608 EC50 = 170 nM T13852 CT57CZ 58329610 EC50 = 6.7 nM T13852 C5YS7U 58329611 EC50 = 0.067 nM T13852 CT3YW4 58329614 EC50 = 83 nM T13852 CWIY64 58329615 EC50 = 3.3 nM T13852 CG2S6C 58329617 EC50 = 25 nM T13852 C30BKS 58390822 EC50 = 2 nM T13852 CMN68P 58390859 EC50 = 0.89 nM T13852 C86MRL 58390878 EC50 = 1.3 nM T13852 CR07UT 58390929 EC50 = 1.1 nM T13852 CD9SZ5 58390949 EC50 = 56 nM T13852 C0X4GY 58390980 EC50 = 1500 nM T13852 C7T0LA 58537167 EC50 = 5 nM T13852 CHU24M 58537193 EC50 = 1.7 nM T13852 CZ6R5C 58537228 EC50 = 0.44 nM T13852 C4IXQ6 58725140 EC50 = 161 nM T13852 CM71ZT 58907531 IC50 = 77 nM T13852 CCJ2B4 58907649 EC50 = 164 nM T13852 CD6EH2 58907658 IC50 = 92 nM T13852 CO26CZ 59146063 EC50 = 5.012 nM T13852 C74YXS 59146106 EC50 < 0.01 nM T13852 CB0IH5 59174152 IC50 = 6.1 nM T13852 C0HN9L 59174265 IC50 = 2.6 nM T13852 CHID06 59176993 EC50 = 12400 nM T13852 C4J3YO 59176995 EC50 = 180 nM T13852 C61FCO 59176999 EC50 = 1800 nM T13852 CG80CT 59177003 EC50 = 8 nM T13852 CGJ30B 59177004 EC50 = 9200 nM T13852 CB7N6D 59177011 EC50 = 1 nM T13852 CI74RQ 59177019 EC50 = 50 nM T13852 C8KVQ9 59177040 EC50 = 650 nM T13852 CU4Y6H 59177057 EC50 = 30 nM T13852 CBIM58 59177061 EC50 = 3 nM T13852 C0PK8M 59177064 EC50 = 310 nM T13852 CEWC27 59177065 EC50 = 7 nM T13852 CB8FD1 59177084 EC50 = 26 nM T13852 C8P7LM 59177085 EC50 = 1000 nM T13852 CCL51E 59177097 EC50 = 190 nM T13852 CMK4G5 59177101 EC50 = 210 nM T13852 C5ZT3B 59177113 EC50 = 12 nM T13852 C8G4ZB 59177115 EC50 = 800 nM T13852 CVP0R2 59177130 EC50 = 1800 nM T13852 C76ZEY 59177131 EC50 = 4000 nM T13852 CI1KY5 59177136 EC50 = 2200 nM T13852 CSI6X5 59177147 EC50 = 23500 nM T13852 C1TKA3 59177155 EC50 = 57 nM T13852 CLD89J 59177166 EC50 = 590 nM T13852 CV4J6H 59177167 EC50 = 2340 nM T13852 C7IK3M 59177172 EC50 = 1170 nM T13852 CWQM60 59177179 EC50 = 5 nM T13852 C1ML6Q 59177180 EC50 = 1840 nM T13852 C3CM8P 59177194 EC50 = 430 nM T13852 CPRZ17 59177196 EC50 = 9000 nM T13852 C1IV9W 59177203 EC50 = 420 nM T13852 CHG68Z 59177207 EC50 = 5 nM T13852 C5SCA8 59177212 EC50 = 800 nM T13852 CNE3U0 59177226 EC50 = 240 nM T13852 CH1BZ8 59177239 EC50 = 27 nM T13852 CO3N7S 59177244 EC50 = 6 nM T13852 CAXI98 59177248 EC50 = 24 nM T13852 CTW94J 59177290 EC50 = 34 nM T13852 CC8PX3 59177293 EC50 = 1100 nM T13852 C38MAI 59202018 EC50 = 7.7 nM T13852 CY2M9Z 59202022 EC50 = 4.3 nM T13852 C9K4HI 59218029 EC50 = 210 nM T13852 C8FZ4S 59384310 EC50 = 0.26 nM T13852 CQ52OA 59384375 EC50 = 0.44 nM T13852 CYF39N 59438732 EC50 = 1830 nM T13852 C7FZ2T 59438736 EC50 = 6340 nM T13852 C7HBW2 59438740 EC50 = 6190 nM T13852 CF62HR 59438762 EC50 = 3170 nM T13852 CF8GJ1 59438788 EC50 = 3230 nM T13852 C9IA0U 59438798 EC50 = 22100 nM T13852 C6UX5A 59438807 EC50 = 2250 nM T13852 CFV31Q 59438811 EC50 = 7690 nM T13852 CZMR84 59438820 EC50 = 2370 nM T13852 CYJ29H 59438827 EC50 = 460 nM T13852 CDA7S4 59451739 IC50 = 5260 nM T13852 CV3RJ6 59451743 IC50 = 6230 nM T13852 CE47JS 59451750 IC50 = 4170 nM T13852 C3D4EZ 59451753 IC50 = 7210 nM T13852 C1CYE5 59451764 IC50 = 1180 nM T13852 CF5VO8 59451770 IC50 = 3030 nM T13852 C7L4SK 59451793 IC50 = 109 nM T13852 CC9FN3 59451797 IC50 = 4410 nM T13852 CQ23ZL 59451812 IC50 = 1780 nM T13852 CU83BX 59451813 IC50 = 656 nM T13852 CLQ46R 59451819 IC50 = 401 nM T13852 C7CR6Z 59451824 IC50 > 10000 nM T13852 CB9S0P 59451832 IC50 > 10000 nM T13852 CRE85M 59451845 IC50 = 220 nM T13852 C0KJ1F 59451849 IC50 = 472 nM T13852 CV94QR 59451859 IC50 > 10000 nM T13852 CR62AY 59451867 IC50 = 9810 nM T13852 CCAI45 59451870 IC50 = 3460 nM T13852 CVY6T4 59451878 IC50 = 3870 nM T13852 CVN69I 59451883 IC50 = 2 nM T13852 C2QZ8N 59495631 Ki = 0.8 nM T13852 CJA5S6 59548622 EC50 = 5.012 nM T13852 CTWM17 59549234 EC50 = 3.2 nM T13852 C8J6GQ 59593534 EC50 = 17.8 nM T13852 CE37MO 59982944 EC50 = 0.3 nM T13852 C4MZP6 60150588 EC50 = 3.4 nM T13852 C1C8SV 60150616 EC50 = 4 nM T13852 C07EBJ 66561414 EC50 = 0.631 nM T13852 C6WM1N 66636736 EC50 = 4.7 nM T13852 CPON94 66636757 EC50 = 0.9 nM T13852 CF59YL 66636847 EC50 = 0.6 nM T13852 C7YA0P 66655198 EC50 = 5011.87 nM T13852 CMT3L8 66655210 EC50 > 10000 nM T13852 C1M4BX 66655282 EC50 = 6309.57 nM T13852 CD09QP 66655362 EC50 = 1584.89 nM T13852 CTX2M1 66655578 EC50 > 31622.78 nM T13852 CASW54 66655584 EC50 = 6309.57 nM T13852 CN83CO 66655586 EC50 = 12589.25 nM T13852 CJG3A2 66655632 EC50 > 31622.78 nM T13852 CI5KQ1 66655655 EC50 > 31622.78 nM T13852 CRGW91 66655753 EC50 = 1584.89 nM T13852 C9PGA0 66655774 EC50 = 1000 nM T13852 C7WVE9 66655956 EC50 = 6309.57 nM T13852 CZS20N 66655962 EC50 > 31622.78 nM T13852 C6UGD4 66655998 EC50 > 31622.78 nM T13852 CQ0U7L 66656025 EC50 > 10000 nM T13852 CKO1L6 66656274 EC50 > 31622.78 nM T13852 CZS9C7 66829256 EC50 = 0.9 nM T13852 C5E0VD 66829275 EC50 = 0.3 nM T13852 CGI61O 66829279 EC50 = 1.3 nM T13852 C4XNF6 66829308 EC50 = 0.7 nM T13852 C5UTG1 66829311 EC50 = 0.5 nM T13852 CW9UH3 66829334 EC50 = 0.5 nM T13852 C5XDU9 66852776 EC50 = 7.9 nM T13852 C8Q9HN 66853439 EC50 = 5 nM T13852 CCBH03 66853698 EC50 = 54 nM T13852 CG69FE 66923349 EC50 = 135 nM T13852 CD9BG6 66931911 EC50 = 10 nM T13852 CY25VM 66955367 EC50 = 1.1 nM T13852 C8X7CG 66955472 EC50 = 4.2 nM T13852 CHZG64 67009121 IC50 = 32 nM T13852 CWD9E5 67009400 IC50 = 548 nM T13852 CU34IA 67009931 IC50 = 297 nM T13852 CDIY38 67010094 IC50 = 228 nM T13852 CYTQ63 67010164 IC50 > 10000 nM T13852 CF1LH2 67193564 EC50 = 57 nM T13852 CGOE75 67193675 EC50 = 2.6 nM T13852 C19JMK 67193896 EC50 = 3.5 nM T13852 C3QCF7 67195432 EC50 = 4.5 nM T13852 CN2K6J 67195504 EC50 = 0.58 nM T13852 C1CR8J 67195758 EC50 = 6.6 nM T13852 CNO54F 67196129 EC50 = 13 nM T13852 CZ3HJ7 67196477 EC50 = 540 nM T13852 CVRG24 67197502 EC50 = 1.4 nM T13852 C6AZY0 67249162 EC50 = 0.13 nM T13852 CX6SF2 67250226 EC50 = 0.025 nM T13852 CP0K7H 67266022 EC50 = 20 nM T13852 CCJ3R5 67284085 EC50 = 398.11 nM T13852 CT0SQ6 67284109 EC50 = 125.89 nM T13852 CA8W5X 67284479 EC50 = 50.12 nM T13852 C8SMB3 67285906 EC50 = 158.49 nM T13852 CW3JD2 67351486 EC50 = 2.7 nM T13852 C0FH4B 67414717 EC50 = 1.4 nM T13852 CMI48F 67415695 EC50 = 300 nM T13852 CHFX15 67416434 EC50 = 6.6 nM T13852 CVK91L 68192087 EC50 = 21 nM T13852 CS0GZ3 68446124 EC50 = 251.19 nM T13852 C0H4RL 68547259 EC50 = 0.3 nM T13852 CMG53F 68553624 EC50 = 0.2 nM T13852 C2KI7M 68555865 EC50 = 0.1 nM T13852 C4Q3NF 68762699 EC50 = 0.1 nM T13852 CD98MX 68763522 EC50 = 1 nM T13852 CT3PC6 69143493 EC50 = 232 nM T13852 CXZ2A1 69143673 EC50 = 5.8 nM T13852 CS2W7J 69144360 EC50 = 9.8 nM T13852 C8RG2L 69144892 EC50 = 902 nM T13852 CV4OD5 69144893 EC50 = 3110 nM T13852 CF76YV 69144915 EC50 = 15 nM T13852 CQ9N2R 69145858 EC50 = 28.6 nM T13852 CY09OV 69263869 EC50 = 7 nM T13852 CK3LG1 69669192 EC50 = 7.5 nM T13852 CCFQ57 70681006 EC50 = 630.96 nM T13852 CQ27UW 70681007 EC50 = 63.1 nM T13852 C6PG3U 70681008 EC50 = 50.12 nM T13852 C6D9LM 70681009 EC50 = 1.585 nM T13852 CY28VU 70681258 EC50 = 0.03162 nM T13852 CO05FX 70681268 IC50 > 10000 nM T13852 C9UD6M 70681384 EC50 = 1.1 nM T13852 CH42VZ 70681385 EC50 = 3.2 nM T13852 CMZ6I4 70681674 EC50 = 1000 nM T13852 CX26ST 70681687 EC50 = 0.03162 nM T13852 CRQO04 70681688 EC50 = 0.1585 nM T13852 CC3SF4 70681689 EC50 = 10 nM T13852 C30MIN 70681812 EC50 = 700 nM T13852 C8CX6G 70681813 EC50 = 81 nM T13852 CKS42M 70681814 EC50 = 21 nM T13852 CALO30 70681815 EC50 = 180 nM T13852 CE5IP4 70682167 EC50 = 630.96 nM T13852 C94ZQP 70682180 EC50 > 3162.28 nM T13852 C7ZF2R 70682181 EC50 > 3162.28 nM T13852 C7IE8O 70683136 EC50 > 10000 nM T13852 C9CND8 70683137 EC50 = 31.62 nM T13852 CTH29P 70683346 EC50 > 3162.28 nM T13852 CEJ51S 70683347 EC50 = 0.03981 nM T13852 CIOV12 70683348 EC50 = 0.07943 nM T13852 CR03ZG 70683349 EC50 = 6.31 nM T13852 C8BSP9 70683465 EC50 = 90 nM T13852 CZFR46 70683478 EC50 = 1.3 nM T13852 CQ29EW 70683479 EC50 = 11 nM T13852 CQ2O3C 70683480 EC50 = 2.8 nM T13852 CH81TY 70683793 EC50 > 3162.28 nM T13852 CHM21Y 70683794 EC50 = 6.31 nM T13852 CR19FO 70683922 EC50 = 8 nM T13852 CBC65V 70684279 EC50 = 5.012 nM T13852 CA0W3R 70684293 EC50 = 1.995 nM T13852 C1UH9R 70684294 EC50 = 251.19 nM T13852 CK1Z3U 70685208 EC50 = 501.19 nM T13852 CLV2B8 70685209 EC50 = 630.96 nM T13852 CX8HF7 70685210 EC50 = 7.943 nM T13852 CG0B8I 70685211 EC50 = 2511.89 nM T13852 CBZ34D 70685212 EC50 = 1000 nM T13852 CQS7I1 70685573 EC50 = 15 nM T13852 CXBU72 70685582 EC50 = 35 nM T13852 C51SBP 70685583 EC50 = 8 nM T13852 C0ZIF9 70685933 EC50 = 158.49 nM T13852 CZ19QH 70685934 EC50 = 63.1 nM T13852 C7MZQ0 70685935 EC50 = 0.3981 nM T13852 C8L0XD 70685939 EC50 = 0.7943 nM T13852 CXU38H 70686050 EC50 = 390 nM T13852 C2ILY4 70686051 EC50 = 2000 nM T13852 CNI10K 70686052 EC50 = 4 nM T13852 CZY89T 70686053 EC50 = 25 nM T13852 CL35WR 70686431 EC50 = 2511.89 nM T13852 CUI3J9 70686445 EC50 > 3162.28 nM T13852 CL31YJ 70687367 EC50 = 6309.57 nM T13852 CLK95G 70687368 EC50 > 3162.28 nM T13852 CN8Z6V 70687369 EC50 = 79.43 nM T13852 C1BTF0 70687554 EC50 = 13 nM T13852 C6JM8Q 70687592 EC50 = 398.11 nM T13852 CF1CE4 70687715 EC50 = 22 nM T13852 C02SFN 70687728 EC50 = 10 nM T13852 CA7RO8 70687729 EC50 = 5.8 nM T13852 C2XU1Y 70687730 EC50 = 4.1 nM T13852 CCQ97S 70688066 EC50 = 0.3162 nM T13852 COCF48 70688067 EC50 = 125.89 nM T13852 CP3UG2 70688177 EC50 = 38 nM T13852 CQ0ZN8 70688528 EC50 = 1.585 nM T13852 C9I4AK 70688545 EC50 = 25.12 nM T13852 C8Q6YJ 70689430 EC50 = 630.96 nM T13852 CGYX75 70689431 EC50 > 10000 nM T13852 CGPI21 70689432 EC50 = 251.19 nM T13852 CW51BD 70689433 EC50 = 251.19 nM T13852 CTI8V1 70689434 EC50 = 0.3981 nM T13852 CC2G3F 70689616 EC50 = 230 nM T13852 C1RP8W 70689617 EC50 = 68 nM T13852 C0NZM7 70689618 EC50 = 5.4 nM T13852 CC8E7V 70689644 EC50 > 10000 nM T13852 CN8L3T 70689653 IC50 = 286 nM T13852 CLHV45 70689764 EC50 = 54 nM T13852 CG65PK 70689765 EC50 = 25 nM T13852 CCB9W1 70689781 EC50 = 5.5 nM T13852 CNS91B 70689782 EC50 = 5.4 nM T13852 CO8TR9 70690085 EC50 = 1000 nM T13852 CJ5KM4 70690096 EC50 = 0.1 nM T13852 CTM09Q 70690589 EC50 = 31.62 nM T13852 C2KQ0O 70690600 EC50 > 3162.28 nM T13852 C1Z3PW 70690601 EC50 > 3162.28 nM T13852 C4JU6G 70690602 EC50 = 1.995 nM T13852 CR51FQ 70690603 EC50 = 1.259 nM T13852 CIMG07 70691539 EC50 = 1258.93 nM T13852 C13XWD 70691540 EC50 = 3981.07 nM T13852 CY78XU 70691541 EC50 = 251.19 nM T13852 CVH73S 70691745 EC50 = 13 nM T13852 CFV37A 70691746 EC50 = 14 nM T13852 CD9HK6 70691922 EC50 = 4.5 nM T13852 CRV82N 70692232 EC50 = 158.49 nM T13852 CO5G0D 70692233 EC50 > 3162.28 nM T13852 CI01GS 70692234 EC50 > 3162.28 nM T13852 CPIX90 70692235 EC50 = 19.95 nM T13852 CAJ78G 70692236 EC50 = 398.11 nM T13852 C1C0DO 70692237 EC50 = 10 nM T13852 C5PT2V 70692238 EC50 = 125.89 nM T13852 CVOW40 70692256 EC50 = 0.3162 nM T13852 C1FIS9 70692257 EC50 = 1 nM T13852 C9Z5LN 70692258 EC50 = 0.3981 nM T13852 C92JOF 70692370 EC50 = 150 nM T13852 C7UNV3 70692732 EC50 = 3.981 nM T13852 CY68TM 70692743 EC50 = 31.62 nM T13852 C2JFY7 70692744 EC50 = 5.012 nM T13852 CYAS67 70693630 EC50 = 316.23 nM T13852 CIG81N 70693631 EC50 = 630.96 nM T13852 C9V3GW 70693632 EC50 = 1258.93 nM T13852 CO0A1Z 70693633 EC50 > 10000 nM T13852 C0OA7T 70693634 EC50 = 125.89 nM T13852 C3NC8P 70693635 EC50 = 630.96 nM T13852 CT7S1Z 70693636 EC50 = 1.259 nM T13852 CKGI50 70693811 EC50 = 38 nM T13852 CJSX34 70693847 EC50 = 3162.28 nM T13852 COP46G 70693848 EC50 > 10000 nM T13852 CT5J1F 70693975 EC50 = 3.5 nM T13852 C7DFY6 70693976 EC50 = 6 nM T13852 CD6I5X 70694325 EC50 = 0.03162 nM T13852 CT12OX 70694326 EC50 = 1.259 nM T13852 CXIB79 70694327 EC50 = 0.07943 nM T13852 CB7CT3 70694328 EC50 = 0.3981 nM T13852 C76HLN 70694426 EC50 = 39 nM T13852 C8PK5N 70694427 EC50 = 18 nM T13852 C8CGR6 70694773 EC50 = 25.12 nM T13852 C6BVJ0 70694787 EC50 = 125.89 nM T13852 C9GH8V 70694788 EC50 = 398.11 nM T13852 C5ZIQ3 70694789 EC50 = 158.49 nM T13852 CDQ83S 70695740 EC50 = 1000 nM T13852 CQBH21 70695741 EC50 > 10000 nM T13852 CBUZ83 70695742 EC50 = 31.62 nM T13852 CFL2H8 70695743 EC50 = 0.03981 nM T13852 C4YT9N 70695932 EC50 = 6.8 nM T13852 C3EAN4 70695958 EC50 = 398.11 nM T13852 CXJ78C 70696095 EC50 = 300 nM T13852 C9HWE1 70696096 EC50 = 3.4 nM T13852 CW0LC8 70696401 EC50 = 0.02512 nM T13852 CA20YS 70696402 EC50 = 398.11 nM T13852 C6WO5Y 70696411 EC50 = 0.5012 nM T13852 CCF0R3 70696493 EC50 = 15 nM T13852 C7TAW1 70696818 EC50 > 10000 nM T13852 C39WMC 70696819 EC50 > 10000 nM T13852 CO35NY 70696832 EC50 = 630.96 nM T13852 C5ARV6 70696833 EC50 = 5.012 nM T13852 C8SEH5 71450072 IC50 = 2.1 nM T13852 CR4V0T 71450073 IC50 = 3.4 nM T13852 C4NKW2 71450719 EC50 = 9000 nM T13852 CS6H0R 71455442 IC50 = 12 nM T13852 C2XK5N 71456056 EC50 = 6600 nM T13852 CBD8E5 71457219 IC50 = 8.4 nM T13852 CUFK75 71460883 IC50 = 20 nM T13852 C3D2TO 71461488 EC50 = 4500 nM T13852 CMQ9J5 71487023 EC50 > 10000 nM T13852 CQV01F 71487029 EC50 = 1611 nM T13852 C16KJX 71540398 IC50 = 370 nM T13852 CB87GJ 71540499 IC50 = 3000 nM T13852 CL91KM 71664646 EC50 = 0.76 nM T13852 COW49V 71711503 EC50 = 2.65 nM T13852 C6ON8T 71711505 EC50 = 81.74 nM T13852 C72TWZ 71718271 EC50 = 1400 nM T13852 CMH9U0 71719476 EC50 = 1700 nM T13852 CK39OJ 72546270 EC50 = 1104 nM T13852 CL9JQ5 72793715 EC50 = 3 nM T13852 CQ54TG 72793716 EC50 = 3.8 nM T13852 C62HAQ 72793717 EC50 = 97 nM T13852 C58ELP 72793719 EC50 > 10000 nM T13852 C85WKP 72793738 EC50 = 7490 nM T13852 C1SC2N 72793739 EC50 = 7280 nM T13852 CSJ7L9 72793740 EC50 > 10000 nM T13852 CWIK42 72793741 EC50 > 10000 nM T13852 CI0N5T 72793759 EC50 > 10000 nM T13852 CNBK82 72793774 EC50 > 10000 nM T13852 C38DCV 72793775 EC50 = 23.7 nM T13852 COHM70 72793788 EC50 = 6.8 nM T13852 CEG7U8 72793789 EC50 = 2.8 nM T13852 CASW13 72793790 EC50 = 3.5 nM T13852 CHO28L 72793791 EC50 = 3.4 nM T13852 C1Y6MK 72793810 EC50 = 0.7 nM T13852 CJ56PQ 72793811 EC50 = 0.7 nM T13852 C3YQ2R 72793820 EC50 = 34.2 nM T13852 C9D5RT 72793821 EC50 = 37.8 nM T13852 CP2M4D 72793822 EC50 = 1.3 nM T13852 C9K8YM 72793828 EC50 = 1 nM T13852 CJ48WM 73333750 EC50 = 40.9 nM T13852 CHMD43 73774584 EC50 = 51 nM T13852 C6G3YC 76310852 EC50 = 1.1 nM T13852 COQY72 76310992 EC50 = 0.1 nM T13852 C2DB3P 76310993 EC50 = 54 nM T13852 CW48DP 76310994 EC50 = 0.9 nM T13852 C2H9FK 76311230 EC50 = 66.3 nM T13852 C3TGY9 76311231 EC50 = 632 nM T13852 CL6ZD0 76311232 EC50 = 37 nM T13852 CA3L2S 76314472 EC50 = 1.8 nM T13852 CC9W0M 76314473 EC50 = 1.1 nM T13852 C56OGS 76314474 EC50 = 4.6 nM T13852 CEN46O 76314475 EC50 = 11 nM T13852 C8MFO0 76314621 EC50 = 0.2 nM T13852 C68NUF 76314622 EC50 = 0.1 nM T13852 C39OGP 76314623 EC50 = 0.4 nM T13852 C04AUW 76314624 EC50 = 0.2 nM T13852 C7AI9H 76314625 EC50 = 0.1 nM T13852 CHYG50 76314626 EC50 = 248 nM T13852 CWVZ73 76317347 EC50 = 8570 nM T13852 CB9L0F 76318055 EC50 = 4.7 nM T13852 CQ6E1G 76318056 EC50 = 20 nM T13852 C2TL1H 76318057 EC50 = 20 nM T13852 CWC1G2 76318058 EC50 = 0.9 nM T13852 C4O8RP 76318194 EC50 = 1110 nM T13852 CYJ3Z8 76318195 EC50 = 2.1 nM T13852 CH9B3U 76318196 EC50 = 8.4 nM T13852 CF7X8W 76318197 EC50 = 23 nM T13852 CR6H1D 76318198 EC50 = 0.2 nM T13852 CY2CW5 76318199 EC50 = 4.6 nM T13852 CA1I7G 76318200 EC50 = 3.9 nM T13852 C6UDP4 76318445 EC50 = 27 nM T13852 C69WSQ 76318446 EC50 = 85.8 nM T13852 C08KVJ 76321769 EC50 = 6.6 nM T13852 C1CZ0H 76321770 EC50 = 2.4 nM T13852 CLB13F 76321771 EC50 = 860 nM T13852 CKR7X3 76321772 EC50 = 4.7 nM T13852 CJ69NG 76321773 EC50 = 1.3 nM T13852 C87GMQ 76321895 EC50 = 0.1 nM T13852 CB0N9L 76321896 EC50 = 0.2 nM T13852 CGC85U 76321897 EC50 = 89 nM T13852 C2V5AL 76322116 EC50 = 203 nM T13852 CA9V2U 76322117 EC50 = 341 nM T13852 C7UL9Q 76322118 EC50 = 886 nM T13852 CVP6Y8 76322119 EC50 = 66.3 nM T13852 CKUS39 76322127 EC50 = 254 nM T13852 C3NK2P 76322128 EC50 = 329 nM T13852 CQ17WJ 76325392 EC50 = 0.4 nM T13852 C4VG0E 76325528 EC50 = 0.3 nM T13852 C90FKU 76325529 EC50 = 2 nM T13852 CXA1J3 76325530 EC50 = 1.3 nM T13852 C3SDU8 76325531 EC50 = 0.7 nM T13852 C9ZQ3K 76325533 EC50 = 0.2 nM T13852 CGLB78 76325739 EC50 = 89 nM T13852 C54XGU 76325748 EC50 = 35 nM T13852 C8IX9H 76325749 EC50 = 529 nM T13852 CN14OE 76328931 EC50 = 0.4 nM T13852 CE5D9I 76329073 EC50 = 0.9 nM T13852 CMG6Q7 76329074 EC50 = 86 nM T13852 CQ5HF1 76329075 EC50 = 1.8 nM T13852 CX4OA0 76329076 EC50 = 4.4 nM T13852 CNH32U 76329077 EC50 = 23 nM T13852 CO9QF7 76329310 EC50 = 14 nM T13852 CF84JV 76329311 EC50 = 800 nM T13852 C3EKT6 76329326 EC50 = 172 nM T13852 CYP53V 76329327 EC50 = 157 nM T13852 CA7GO0 76332613 EC50 = 79 nM T13852 CI48VM 76332614 EC50 = 1600 nM T13852 CPCU86 76332615 EC50 = 6 nM T13852 CE0U5H 76332741 EC50 = 1 nM T13852 CNI13W 76332955 EC50 = 48.1 nM T13852 CCJ1E9 76332956 EC50 = 52.9 nM T13852 CP4M6B 76332957 EC50 = 932 nM T13852 C5ZW4J 76336211 EC50 = 1.4 nM T13852 COB8X9 76336212 EC50 = 1.6 nM T13852 CNJ13I 76336213 EC50 = 4.8 nM T13852 C0XIK8 76336214 EC50 = 1.3 nM T13852 CFU3C9 76336215 EC50 = 48 nM T13852 CVM60F 76336361 EC50 = 0.3 nM T13852 C1VJZ3 76336362 EC50 = 0.8 nM T13852 CGTV16 76336363 EC50 = 9.5 nM T13852 C0O2NK 76336364 EC50 = 0.1 nM T13852 COX87F 76336566 EC50 = 19.8 nM T13852 C1EZ9S 76336567 EC50 = 876 nM T13852 CB5NI0 76336568 EC50 = 91.5 nM T13852 C42TIC 76336569 EC50 = 72 nM T13852 C9IKU5 78321974 EC50 = 0.006 nM T13852 CK4S8A 86646444 EC50 = 26 nM T13852 CI1WF3 89710483 EC50 = 316.23 nM T13852 C2G1HE 89710485 EC50 = 1258.93 nM T13852 CJ6RC9 89710536 EC50 = 5011.87 nM T13852 CGE95T 89710694 EC50 = 316.23 nM T13852 CLP73T 89710808 EC50 = 1258.93 nM T13852 CR0LX1 89711073 EC50 = 3981.07 nM T13852 C2D4SQ 89713031 EC50 = 125.89 nM T13852 C0TQK5 89713056 EC50 = 316.23 nM T13852 CL74JM 90309142 IC50 > 10000 nM T13852 CY7K8V 91758813 EC50 = 1.7 nM T13852 C3XVO1 101863648 IC50 = 18 nM T13852 C51VMH 118707012 EC50 = 7 nM T13852 C5K8VH 118707193 EC50 = 3 nM T13852 CX1UP2 118707194 EC50 = 19 nM T13852 CEI4M5 118707195 EC50 = 2.8 nM T13852 CKR17A 118707196 EC50 = 4 nM T13852 CA0K5C 118707197 EC50 = 2.3 nM T13852 C9SQ5X 118707198 EC50 = 2.2 nM T13852 CL1EJ7 118707199 EC50 = 6.5 nM T13852 C9C0FB 118716137 EC50 = 685 nM T13852 CQJ87G 118716138 EC50 = 93.9 nM T13852 CMJ7B8 118716139 EC50 = 12.8 nM T13852 C4D5QX 118716140 EC50 = 7.6 nM T13852 CK0C5M 118716141 EC50 = 16.3 nM T13852 C3C6VG 118716142 EC50 = 9.1 nM T13852 C6S5FV 118716143 EC50 = 10.9 nM T13852 CSR50K 118716144 EC50 = 74 nM T13852 CP6W7I 118716145 EC50 = 25.4 nM T13852 C3KN6Y 118716146 EC50 = 22.2 nM T13852 CPR5Y4 118716147 EC50 = 42.4 nM T13852 CH0P9G 118716148 EC50 = 147.6 nM T13852 CA10EJ 118716149 EC50 = 69.5 nM T13852 CM14DZ 118716150 EC50 = 48.9 nM T13852 CG3OD8 118716151 EC50 = 108.2 nM T13852 C8XNF6 118716152 EC50 = 25.8 nM T13852 COIL26 118716153 EC50 = 54.5 nM T13852 C4QBP2 118716154 EC50 = 17.8 nM T13852 C5JTY2 118716155 EC50 = 343 nM T13852 CL78NH 118716156 EC50 = 154 nM T13852 CSP01A 118716157 EC50 = 64.1 nM T13852 C2WY3I 118716177 EC50 = 111 nM T13852 CJ2X5A 118716178 EC50 = 126 nM T13852 C0N6LQ 118716179 EC50 = 1626 nM T13852 CGQ3D4 118716180 EC50 = 42 nM T13852 CI6J2D 118716181 EC50 = 22 nM T13852 COX9P3 118716182 EC50 = 15 nM T13852 C79NHT 118716183 EC50 = 53 nM T13852 CTQO81 118716184 EC50 = 29 nM T13852 C3L2JK 118716185 EC50 = 19 nM T13852 C0AK1I 118716186 EC50 = 257 nM T13852 CV2NB9 118716187 EC50 = 1287 nM T13852 C86HJL 118716188 EC50 = 638 nM T13852 C5T1DG 118716189 EC50 = 630 nM T13852 CJ0PM8 118716190 EC50 = 551 nM T13852 CB25DV 118717764 EC50 = 3.1 nM T13852 CH43DI 118717765 EC50 = 1300 nM T13852 CV8IT1 118717766 EC50 = 17 nM T13852 CT3U1D 118717767 EC50 = 46 nM T13852 CXS94P 118717768 EC50 = 3600 nM T13852 C41LOQ 118717769 EC50 = 420 nM T13852 CP1VA0 118717770 EC50 = 1.2 nM T13852 C2HTU4 118717771 EC50 = 9.8 nM T13852 CRS38A 118717772 EC50 = 6.5 nM T13852 CJC90W 118717773 EC50 = 4.1 nM T13852 CFH74U 118717774 EC50 = 2400 nM T13852 C5NVP7 118717775 EC50 = 92 nM T13852 CH7OB1 118717776 EC50 = 5.3 nM T13852 CPG9M3 118717777 EC50 = 0.5 nM T13852 CK2L1R 118717778 EC50 = 2.3 nM T13852 CS62RG 118717779 EC50 = 55 nM T13852 CHV80J 118717780 EC50 = 45 nM T13852 C5QG8O 118717781 EC50 = 12 nM T13852 C3BX4H 118717782 EC50 = 1600 nM T13852 CIKX78 118717783 EC50 > 10000 nM T13852 CT85QI 118717784 EC50 > 5400 nM T13852 C69IKB 118717785 EC50 = 1100 nM T13852 C6XA2I 118717786 EC50 = 910 nM T13852 C9GN1O 118717787 EC50 = 1100 nM T13852 CQ8E5P 118717788 EC50 = 1100 nM T13852 C5JVO1 118717789 EC50 = 1200 nM T13852 CW7Y8V 118717790 EC50 > 10000 nM T13852 CLXR38 118717791 EC50 > 10000 nM T13852 CW5XJ2 118717792 EC50 = 2700 nM T13852 CA6N4E 118717793 EC50 = 240 nM T13852 CS4V1Q 118717794 EC50 = 2100 nM T13852 CV83BZ 118717795 EC50 = 0.5 nM T13852 C83CMX 118723170 EC50 = 120 nM T13852 C6Y0VB 118723864 EC50 = 6.31 nM T13852 CK23TG 118724202 EC50 = 31.62 nM T13852 CFL73Q 118724203 EC50 = 19.95 nM T13852 C72NCP 118728432 IC50 > 10000 nM T13852 CRMI76 118729154 EC50 = 340 nM T13852 CGC41A 118729155 EC50 = 2690 nM T13852 C9MU7D 118729156 EC50 > 100000 nM T13852 CI4UD7 118729157 EC50 = 220 nM T13852 CV2WQ5 118729158 EC50 = 490 nM T13852 CC30FH 118729159 EC50 = 670 nM T13852 C7YNG9 118729160 EC50 = 15200 nM T13852 CA96UT 118729161 EC50 > 100000 nM T13852 C6L3GO 118729162 EC50 = 410 nM T13852 CXZP24 118729163 EC50 = 250 nM T13852 C4KR9I 118729164 EC50 > 33000 nM T13852 CG2U1Z 118729920 EC50 = 170 nM T13852 C9WIF6 118729921 EC50 = 1.4 nM T13852 CU0C1S 122186560 EC50 = 9 nM T13852 CCWG18 122186561 EC50 = 130 nM T13852 CI1Y7B 122186562 EC50 = 2420 nM T13852 CH23UV 124171442 EC50 = 42 nM T13852 C9VT4Z 124171444 EC50 = 11 nM T13852 CX8VT2 124171447 EC50 = 50 nM T13852 CONE63 124171453 EC50 = 32 nM T13852 CPJU69 124171486 EC50 = 0.1 nM T13852 C5U6VC 124171493 EC50 = 67 nM T13852 CPL30Z 124171494 EC50 = 49 nM T13852 C4P9IE 124171496 EC50 = 0.5 nM T13852 CE8C9A 124171498 EC50 = 4.1 nM T13852 C9ADH2 124171513 EC50 = 62 nM T13852 CCOE71 124173029 EC50 = 594 nM T13852 C0VG1S 124173030 EC50 = 105 nM T13852 C4OU5P 124173031 EC50 = 130 nM T13852 CN3K4Z 124173226 EC50 = 18 nM T13852 CD3YQ7 124173228 EC50 = 0.8 nM T13852 C6LQV1 124173275 EC50 = 13 nM T13852 C9U4QR 124221654 EC50 > 100000 nM T13852 CE6YZ3 127025658 EC50 = 63.1 nM T13852 CZLV05 127026555 EC50 > 31622.78 nM T13852 CY1HK0 127026677 EC50 = 13 nM T13852 CP2OX6 127027154 EC50 = 251.19 nM T13852 CN0O5K 127028145 EC50 > 31622.78 nM T13852 C17NBX 127028146 EC50 = 6309.57 nM T13852 CQ48GC 127028147 EC50 = 2511.89 nM T13852 C3WM4Z 127028148 EC50 = 1584.89 nM T13852 CIRY67 127028149 EC50 = 3981.07 nM T13852 CN17JT 127028150 EC50 = 1258.93 nM T13852 C6XK7V 127028151 EC50 = 251.19 nM T13852 CF3YN0 127028156 EC50 = 100 nM T13852 CL5IF7 127028461 EC50 = 501.19 nM T13852 C95FHV 127028462 EC50 = 1000 nM T13852 C1LJ2E 127028463 EC50 = 125.89 nM T13852 CDQ8X2 127028464 EC50 = 251.19 nM T13852 C63BMS 127028465 EC50 = 251.19 nM T13852 C01GPK 127029098 EC50 = 25118.86 nM T13852 CIM27T 127029099 EC50 = 1000 nM T13852 CPT32H 127029100 EC50 = 19.95 nM T13852 C0WPV4 127029101 EC50 = 2511.89 nM T13852 CQT30N 127029102 EC50 = 10000 nM T13852 CC4ZH2 127029506 EC50 = 4 nM T13852 C7QMK2 127032587 EC50 = 7 nM T13852 C6W7TO 127032588 EC50 > 10000 nM T13852 CREP02 127032589 EC50 = 13.3 nM T13852 CI51JP 127034581 EC50 = 1524 nM T13852 C0IE2P 127034810 EC50 = 147 nM T13852 CA7SR9 127035166 EC50 = 20 nM T13852 CJ3FN4 127035167 EC50 = 86 nM T13852 CE8Q6D 127036057 EC50 = 0.6 nM T13852 CM31OG 127036062 EC50 = 330 nM T13852 CUI1W5 127036194 EC50 = 4.1 nM T13852 C2DI8M 127036240 EC50 = 560 nM T13852 CD8U3G 127036241 EC50 = 3.5 nM T13852 CW0J4D 127036242 EC50 = 250 nM T13852 C8AX9V 127036243 EC50 = 6 nM T13852 C17ZTC 127036244 EC50 = 0.8 nM T13852 CYPZ61 127036262 EC50 = 0.5 nM T13852 CBK2N7 127036263 EC50 = 2.8 nM T13852 C9IBW0 127036403 EC50 = 120 nM T13852 C6ZS0R 127036404 EC50 = 7.9 nM T13852 C0BVN2 127036405 EC50 = 37 nM T13852 CKRA31 127036406 EC50 = 18 nM T13852 CXI8Z4 127036425 EC50 = 63 nM T13852 CA2OL8 127036426 EC50 = 7.3 nM T13852 C4RPC8 127036427 EC50 = 1.4 nM T13852 C3J0WL 127036428 EC50 = 150 nM T13852 C3JK9E 127036429 EC50 = 200 nM T13852 C4Y7QU 127036430 EC50 = 2.5 nM T13852 C85ZHQ 127036459 EC50 = 310 nM T13852 CDK60U 127037053 EC50 = 550 nM T13852 CJKF28 127037054 EC50 = 14 nM T13852 CJR72C 127037055 EC50 = 300 nM T13852 COCN58 127037056 EC50 = 0.8 nM T13852 C67ADW 127037195 EC50 = 160 nM T13852 CZXY49 127037196 EC50 = 0.2 nM T13852 C76FJO 127037451 EC50 = 0.8 nM T13852 CL70FK 127037694 IC50 = 18 nM T13852 CQ37LX 127037695 IC50 = 5 nM T13852 CM54QV 127037696 IC50 = 48 nM T13852 CD52GS 127041987 IC50 = 2 nM T13852 CG90DH 127045708 EC50 = 1.3 nM T13852 CT2FY0 127045962 EC50 = 6.4 nM T13852 CN8Y5X 127045963 EC50 = 14 nM T13852 C0WDZ1 127046095 EC50 = 310 nM T13852 C1HW3J 127046096 EC50 = 97 nM T13852 CXM68P 127046097 EC50 = 2350 nM T13852 CNVH82 127046130 EC50 = 44 nM T13852 C1FPU6 127046179 EC50 = 55 nM T13852 CR6H8S 127046182 EC50 = 25 nM T13852 C9QXJ5 127046183 EC50 = 28 nM T13852 C7XSZ6 127046184 EC50 = 0.2 nM T13852 C91DCL 127046185 EC50 = 0.3 nM T13852 C6PU3Y 127046323 EC50 = 69 nM T13852 CDKY27 127046324 EC50 = 230 nM T13852 CX38TU 127046325 EC50 = 1 nM T13852 CE2O1K 127046399 EC50 = 0.7 nM T13852 C63EGK 127046400 EC50 = 1.1 nM T13852 CG06MF 127046456 EC50 = 15 nM T13852 C6CZ1K 127046548 EC50 = 0.3 nM T13852 C09FWP 127046549 EC50 = 0.7 nM T13852 CHQ87M 127046550 EC50 = 1.5 nM T13852 CG90HA 127046551 EC50 = 21 nM T13852 CPV3A5 127046566 EC50 = 4.5 nM T13852 CLS7H0 127046567 EC50 = 1 nM T13852 CR25DJ 127046568 EC50 = 11 nM T13852 CVRA82 127046640 EC50 = 190 nM T13852 CT1U5D 127046641 EC50 = 305 nM T13852 CL5PG6 127046741 EC50 = 1 nM T13852 C83BTN 127046742 EC50 = 1.1 nM T13852 CPB61O 127046743 EC50 = 1.1 nM T13852 CH6W9G 127046863 EC50 = 189 nM T13852 CA40VG 127046864 EC50 = 293 nM T13852 C3RCI0 127046865 EC50 = 5.4 nM T13852 CNX35J 127046866 EC50 = 6.8 nM T13852 C1M3IE 127046992 EC50 = 50 nM T13852 C05PXK 127047020 EC50 = 0.3 nM T13852 C76SEA 127047083 EC50 = 0.6 nM T13852 C7WS0V 127047084 EC50 = 1.4 nM T13852 C63NVZ 127047144 EC50 = 270 nM T13852 C9J1HQ 127047145 EC50 = 2090 nM T13852 C5CSZ1 127047225 EC50 = 203 nM T13852 C1PFQ4 127047226 EC50 = 160 nM T13852 CY5O0B 127047690 EC50 = 490 nM T13852 CCEF35 127047778 EC50 = 230 nM T13852 C4KL3G 127047779 EC50 = 285 nM T13852 C0Y3WZ 127047780 EC50 = 305 nM T13852 CB43PM 127047986 EC50 = 385 nM T13852 CHC04K 127048099 EC50 = 2.8 nM T13852 CP91CD 127048100 EC50 = 155 nM T13852 CYDJ81 127048101 EC50 = 14 nM T13852 C7L2PZ 127048102 EC50 = 45 nM T13852 CU1I7S 127048103 EC50 = 110 nM T13852 CM9L1X 127048104 EC50 = 40 nM T13852 CO0I8C 127048141 EC50 = 8.5 nM T13852 C25KAZ 127048142 EC50 = 3.2 nM T13852 CDZ3C4 127048143 EC50 = 4.3 nM T13852 CR47MS 127048144 EC50 = 95 nM T13852 CUE0N7 134130169 EC50 > 100000 nM T13852 C3NC1O 134130546 EC50 > 100000 nM T13852 CJH4K9 134130548 EC50 > 100000 nM T13852 C6JB4Z 134130695 EC50 > 100000 nM T13852 C6V4DA 134130884 EC50 > 100000 nM T13852 CNVC46 134131381 EC50 > 100000 nM T13852 CRB05V 134319250 EC50 = 20 nM T13852 C2JQ7P 134319251 EC50 = 130 nM T13852 C2KHY7 134319262 EC50 = 12 nM T13852 CSK4I8 134319263 EC50 = 10 nM T13852 CUH3P6 134319264 EC50 = 19 nM T13852 C8ZX0N 134319265 EC50 = 30 nM T13852 CRS09O 134319702 EC50 = 1 nM T13852 CZ8MH2 136053659 EC50 = 630.96 nM T13852 CR7Z3E 136147416 EC50 = 16 nM T13852 C2CHL4 137638716 IC50 = 7.7 nM T13852 C81HEI 137644547 Ki = 2.9 nM T13852 C42VXM 137646436 EC50 = 15 nM T13852 CAJY69 137651211 IC50 = 12 nM T13852 C25TZL 137655932 IC50 = 8.4 nM T13852 CH2AN7 137660780 IC50 > 10000 nM T13852 CHRG61 145964044 EC50 > 31622.78 nM T13852 C0ZM4R 145966230 IC50 > 1000 nM T13852 CR8Q4L 145969830 EC50 > 31622.78 nM T13852 CN8IE0 145975394 EC50 = 1995.26 nM T13852 C6JW8K 145976329 IC50 > 1000 nM T13852 C7MI9V 145978086 EC50 = 251.19 nM T13852 CNO90A 145979230 IC50 = 2.512 nM T13852 CD1ZB9 145986468 IC50 = 125.89 nM T13852 C08NSZ 145989628 IC50 > 1000 nM T13852 CH9WB2 145989943 IC50 > 1000 nM T13852 CWT6S7 145990307 IC50 = 316.23 nM T13852 CW38AH 145991829 IC50 = 100 nM T13852 C0T8SM 145993059 IC50 > 1000 nM T13852 CRF7V0 155317229 IC50 > 1000 nM T13852 CX76PB 155317261 IC50 > 1000 nM T13852 CW10AC 155317265 IC50 > 1000 nM T13852 C43CXP 155317276 IC50 > 1000 nM T13852 CLG86C 155317279 IC50 > 1000 nM T13852 CC17FU 155513062 EC50 = 12 nM T13852 CD73QT 155522973 IC50 = 1.8 nM T13852 CI3BA5 155527137 EC50 = 230 nM T13852 C9I7SA 155528529 EC50 = 7.8 nM T13852 CL0E5D 155534250 IC50 = 0.51 nM T13852 CE4W7D 155537600 EC50 = 9.7 nM T13852 C29FQW 155537818 IC50 = 1.5 nM T13852 C37AGW 155538268 EC50 = 2.4 nM T13852 C78VOU 155542034 EC50 = 7.8 nM T13852 CI4X9B 155543631 EC50 = 3.9 nM T13852 CH28SZ 155550350 IC50 = 0.13 nM T13852 CPY85W 16215109 EC50 > 1000 nM T13852 CZSI05 44438257 EC50 > 1000 nM T13852 CWKU57 44438259 EC50 > 1000 nM T13852 CT3AX1 44438261 EC50 > 1000 nM T13852 D00VHN 46905530 IC50 = 0.28 nM T13852 D02LTS 59393720 IC50 = 2 nM T13852 D03AAC 6857802 Ki = 18 nM T13852 D03BRM 11259583 EC50 = 1.2 nM T13852 D04IAF 11452022 EC50 = 0.006 nM T13852 D04XCB 10149595 IC50 = 1900 nM T13852 D05EDD 11588811 EC50 = 58 nM T13852 D05KEE 10904818 EC50 = 0.7943 nM T13852 D06DYN 9908268 EC50 = 0.005 nM T13852 D06GFH 11545181 Ki = 30 nM T13852 D06XMB 44394220 IC50 = 23 nM T13852 D07EAB 10215259 IC50 = 20 nM T13852 D08VLT 10125714 IC50 = 710 nM T13852 D08ZYC 11595431 EC50 < 31622.78 nM T13852 D0D5QS 11725751 IC50 = 3.1 nM T13852 D0LO4T 10287034 IC50 = 0.33 nM T13852 D0N0BN 44394248 IC50 = 360 nM T13852 D0P1TY 44344193 IC50 = 2.3 nM T13852 D0P2AZ 10149721 IC50 = 18 nM T13852 D0ZU0O 4077460 EC50 = 13 nM T86573 D06IAR 60961 Ki > 100000 nM T86573 D0F0ZE 153241 IC50 = 10 nM T86573 CEA89F 10256 IC50 = 22700 nM T86573 C8IOM3 230282 IC50 = 20900 nM T86573 C5ZC0A 497770 IC50 = 20 nM T86573 C4U0OC 497771 IC50 = 25 nM T86573 CLO3N7 497772 IC50 = 70 nM T86573 C4A6KW 497773 IC50 = 85 nM T86573 C0O2NT 497774 IC50 = 23 nM T86573 C2Z5CN 497775 IC50 = 97 nM T86573 CI1L3Y 497776 IC50 = 115 nM T86573 CG2VI5 497777 IC50 = 127 nM T86573 CBD46Q 497781 IC50 = 27 nM T86573 C15XDV 497782 IC50 = 86 nM T86573 CZ8C9D 497783 IC50 = 30 nM T86573 CPJZ06 497784 IC50 = 18 nM T86573 CY06OL 497785 IC50 = 22 nM T86573 CE3SV8 497786 IC50 = 15 nM T86573 C9O4ES 497787 IC50 = 17 nM T86573 C19KSA 497788 IC50 = 13 nM T86573 C6V0PS 497790 IC50 = 11 nM T86573 C25GVM 497791 IC50 = 13 nM T86573 C1RCH0 497792 IC50 = 12 nM T86573 CSR10C 510912 IC50 = 19 nM T86573 C5NK2J 510914 IC50 > 10000000 nM T86573 CMH8E2 510915 IC50 = 670 nM T86573 CRA21X 510916 IC50 = 230 nM T86573 CZU3J2 510917 IC50 > 5000000 nM T86573 C42PBY 510918 IC50 = 33 nM T86573 C85EAF 510919 IC50 = 440 nM T86573 C8S1IN 510920 IC50 = 490 nM T86573 CTG6D2 510921 IC50 > 550 nM T86573 CFM70Y 510923 IC50 = 280 nM T86573 C8WB2K 510924 IC50 = 180 nM T86573 CZK7N2 510925 IC50 = 260 nM T86573 C7BXI5 510926 IC50 = 200 nM T86573 CT78CW 510927 IC50 = 130 nM T86573 CH65RZ 510928 IC50 = 100 nM T86573 C89EVQ 510929 IC50 = 94 nM T86573 CDX01M 510930 IC50 = 180 nM T86573 CTA12W 510933 IC50 = 240 nM T86573 CY8NB9 510934 IC50 = 420 nM T86573 CZ8B4H 510935 IC50 = 210 nM T86573 CA8V3T 588991 IC50 > 5000 nM T86573 C0BCA8 612046 IC50 > 5000 nM T86573 C1K4GB 675297 IC50 >= 5000 nM T86573 C8WTH9 776662 IC50 >= 5000 nM T86573 COJ29X 890649 IC50 = 2100 nM T86573 CQC02U 1139867 IC50 > 5000 nM T86573 CLQ93F 1256741 IC50 > 5000 nM T86573 CO48PU 1367213 IC50 > 5000 nM T86573 CUK93P 2309238 IC50 >= 5000 nM T86573 CK47YQ 2336594 IC50 >= 5000 nM T86573 CM2G8F 2349729 IC50 > 5000 nM T86573 C7TZ5D 2930546 IC50 = 5700 nM T86573 C9A5GP 2953497 IC50 > 5000 nM T86573 CC69EB 2953546 IC50 > 5000 nM T86573 CS1OL3 2990648 IC50 > 5000 nM T86573 C70OXL 3006288 Ki = 3000 nM T86573 CF8N3B 3140491 EC50 > 50000 nM T86573 CAY86S 3312427 IC50 = 2100 nM T86573 CC7WN4 3984960 IC50 > 5000 nM T86573 C0CX1O 4084632 IC50 > 5000 nM T86573 C7KV2M 5173303 IC50 > 5000 nM T86573 CIXQ25 6478685 IC50 = 1400 nM T86573 CW62YA 6479888 IC50 = 790 nM T86573 CN29OD 6618978 IC50 > 50000 nM T86573 CQ96MK 9400179 IC50 > 5000 nM T86573 C75FLA 9797026 IC50 = 10 nM T86573 CND1O9 9797707 IC50 = 190 nM T86573 CJ29KX 9798978 IC50 = 47 nM T86573 C6KM5A 9817941 IC50 = 18.6 nM T86573 CW84FQ 9819013 IC50 = 19 nM T86573 CWC79A 9822362 IC50 < 5 nM T86573 CI8K7N 9838854 IC50 = 5 nM T86573 CLIF21 9842306 IC50 = 23 nM T86573 C0TUD2 9856426 IC50 = 110 nM T86573 CM73SE 9858793 IC50 < 5 nM T86573 CRLZ80 9878581 IC50 = 220 nM T86573 CGB78L 9880305 IC50 = 9 nM T86573 CW3S9G 9883477 Ki = 7 nM T86573 C0S2OY 9884816 IC50 > 10000 nM T86573 CKY2D7 9901690 IC50 = 55 nM T86573 CW4DN6 9906308 IC50 = 150 nM T86573 CG16TY 9907596 IC50 = 30 nM T86573 C64CDR 9912093 IC50 = 20 nM T86573 C4B2QY 9913339 IC50 = 17 nM T86573 CWR2S7 9921131 IC50 = 300 nM T86573 C7HBG3 9921906 IC50 = 200 nM T86573 CK13BM 9923286 IC50 = 63 nM T86573 C5LZ0F 9939667 IC50 = 2600 nM T86573 CO6CV0 9946220 IC50 = 1500 nM T86573 C2H4YG 9947722 IC50 = 14 nM T86573 C4F9QU 9949504 IC50 = 240 nM T86573 CYOD07 9949676 IC50 = 52 nM T86573 CYU51P 9966370 IC50 = 32 nM T86573 CV68RP 9966794 IC50 = 70 nM T86573 CN59SI 9976927 IC50 = 300 nM T86573 CNU0B4 10113643 IC50 < 5 nM T86573 CYM8X2 10117522 IC50 = 68 nM T86573 CI06PF 10126668 IC50 = 130 nM T86573 C49BEK 10131333 IC50 = 34 nM T86573 CG53VS 10131739 IC50 = 18 nM T86573 C0XAE4 10131741 IC50 = 320 nM T86573 C3G5HN 10134808 IC50 = 12 nM T86573 CA6V7K 10135675 IC50 = 55 nM T86573 C9G7LN 10136663 IC50 = 16 nM T86573 CUA05R 10136713 IC50 = 14 nM T86573 CLN19D 10159708 IC50 = 18 nM T86573 C6ELS3 10164678 IC50 = 18 nM T86573 CF9X7W 10172305 IC50 = 86 nM T86573 C2T1ZL 10177736 IC50 = 30 nM T86573 C7Y0NW 10180910 IC50 = 13 nM T86573 CE6F2O 10182966 IC50 = 12 nM T86573 C2O5AZ 10194459 IC50 = 390 nM T86573 CS7W5A 10200804 IC50 = 22 nM T86573 C7MY4A 10203029 IC50 = 15 nM T86573 CR1N6A 10215650 IC50 = 57 nM T86573 CQT82I 10221809 IC50 = 25 nM T86573 CR59ZE 10225421 IC50 = 20 nM T86573 C2X6TP 10233633 Ki = 380 nM T86573 CN4V6E 10236318 IC50 = 104 nM T86573 C05NVJ 10259194 Ki = 300 nM T86573 CW49NI 10269167 IC50 = 2200 nM T86573 CK4L2E 10269960 IC50 = 1100 nM T86573 C87NBG 10270744 IC50 = 28 nM T86573 C48IXR 10273163 IC50 = 6 nM T86573 CN0CM7 10276405 IC50 < 5 nM T86573 CC7PU9 10292172 IC50 = 280 nM T86573 C5OGE6 10297318 IC50 = 11 nM T86573 CLO3B8 10309152 IC50 = 188 nM T86573 CD4L2P 10309428 IC50 = 160 nM T86573 CGF36N 10315709 IC50 < 5 nM T86573 C7IQE9 10323922 IC50 = 16 nM T86573 CV7RA9 10338010 IC50 = 400 nM T86573 CH74QD 10345767 IC50 = 40 nM T86573 CO3GQ6 10358016 IC50 = 28 nM T86573 CU8C2Y 10358687 IC50 = 57 nM T86573 CNG97X 10361468 IC50 = 440 nM T86573 C5WXT0 10381198 IC50 = 12.6 nM T86573 COT86A 10412176 IC50 = 58 nM T86573 CDXB75 10434905 IC50 = 7 nM T86573 C49WRJ 10462123 IC50 = 700 nM T86573 C28SEY 10492850 IC50 = 51800 nM T86573 CF3D8K 10495354 IC50 = 33.5 nM T86573 C7BS3V 10495605 IC50 = 8.51 nM T86573 C02SWN 10496064 IC50 = 465 nM T86573 C6GK2Y 10497453 IC50 = 1800 nM T86573 C0MRX3 10515627 IC50 > 100000 nM T86573 C6MY4S 10518087 IC50 = 537 nM T86573 CPC4F9 10519658 IC50 = 244 nM T86573 CC3HM6 10519938 IC50 = 184 nM T86573 CB5SI1 10544613 IC50 = 231 nM T86573 C7KPV1 10546858 IC50 = 130 nM T86573 C8M9IK 10566972 IC50 = 1700 nM T86573 C37FNC 10567307 IC50 = 437 nM T86573 CFN5V6 10568712 IC50 = 644 nM T86573 CXMB45 10569189 IC50 = 795 nM T86573 C8WM7C 10590744 IC50 = 515 nM T86573 CV4A8H 10593915 IC50 > 100000 nM T86573 C0AWD9 10616470 IC50 = 557 nM T86573 CXE6C1 10637391 IC50 = 959 nM T86573 C06DYP 10643207 IC50 = 1040 nM T86573 C71JXF 10652408 Ki = 270 nM T86573 C2S6QL 10662964 IC50 = 2880 nM T86573 C1CFT4 10663129 IC50 = 15500 nM T86573 CUGI51 10682843 IC50 = 90800 nM T86573 C56XFB 10685057 IC50 = 50000 nM T86573 C50IUC 10686776 IC50 = 11800 nM T86573 CR0MC9 10687933 IC50 > 100000 nM T86573 C5H9AV 10688491 IC50 = 763 nM T86573 CDY41T 10709084 IC50 = 69.3 nM T86573 CMV3K1 10709184 IC50 = 1380 nM T86573 C1S4LW 10709494 IC50 = 14800 nM T86573 C1N0ZQ 10709767 IC50 = 1120 nM T86573 CA7IP0 10709955 IC50 = 52300 nM T86573 CEI9K7 10710928 IC50 = 681 nM T86573 CSW57G 10711760 IC50 = 410 nM T86573 C9S8WO 10713240 IC50 = 462 nM T86573 C87BPJ 10732226 IC50 = 6960 nM T86573 CA4L7V 10735580 IC50 = 126 nM T86573 C0PL3X 10735599 IC50 = 121 nM T86573 CLYM27 10746991 Ki = 320 nM T86573 C8A4YB 10756343 IC50 = 1080 nM T86573 CTSY82 10757447 IC50 = 489 nM T86573 CA4S3R 10758796 IC50 = 50.7 nM T86573 COG9Z8 10759053 IC50 > 100000 nM T86573 C39CHI 10759638 IC50 = 620 nM T86573 CR2A8D 10780300 IC50 = 18800 nM T86573 C1RX9K 10782926 IC50 = 420 nM T86573 C0IM7L 10787380 IC50 = 592 nM T86573 CB4YR2 10803200 IC50 = 1600 nM T86573 CSCY60 10804648 IC50 = 1220 nM T86573 CPU5G1 10805499 IC50 = 140 nM T86573 C9ZU8R 10826397 IC50 = 17000 nM T86573 CR83PV 10826452 IC50 > 100000 nM T86573 C5WAI9 10828540 IC50 = 289 nM T86573 CJ4S2P 10832148 IC50 = 36.7 nM T86573 CDT59Z 10841975 Ki = 57900 nM T86573 CB92AM 10851956 IC50 = 534 nM T86573 C0OIC1 10852317 IC50 = 11900 nM T86573 CQHG03 10872836 IC50 = 104 nM T86573 CO1V7B 10896057 IC50 = 20 nM T86573 C9KVM0 10927586 IC50 = 141 nM T86573 CT8DX2 11069304 Ki = 400 nM T86573 CD4JG6 11118869 IC50 = 254 nM T86573 CAL6D3 11162210 IC50 >= 5000 nM T86573 CR5J2F 11440390 IC50 = 13 nM T86573 C0US3F 11670037 IC50 = 35 nM T86573 C3XHB6 11674857 IC50 = 76 nM T86573 C17DLS 11828231 Ki = 470 nM T86573 C58ZYV 11962096 IC50 = 84 nM T86573 C6IMB3 12093478 IC50 = 970 nM T86573 C54TFI 12093480 IC50 = 110 nM T86573 CGT24F 12093481 IC50 = 73 nM T86573 CLP6T3 15040652 IC50 > 5000 nM T86573 C1N8XS 16007061 IC50 = 13 nM T86573 C4RKU7 16046198 Ki = 37 nM T86573 CKTA70 16484765 IC50 = 2600 nM T86573 CH0R7U 16484780 IC50 = 3200 nM T86573 CN5AB6 16747704 Ki = 18800 nM T86573 C94FVH 16748017 IC50 = 19 nM T86573 C47PSG 16748018 IC50 = 95 nM T86573 CK75MC 16748019 IC50 = 53 nM T86573 CZEQ54 16748020 IC50 = 42 nM T86573 C56GJV 16748021 IC50 = 11 nM T86573 CF85SK 16748022 IC50 = 11 nM T86573 C81DQT 16748142 IC50 = 12 nM T86573 C93QIS 16748143 IC50 = 7.9 nM T86573 C0JYU6 16748144 IC50 = 23 nM T86573 CI3DJ9 16748145 IC50 = 14 nM T86573 CA6M0N 16748267 IC50 = 12 nM T86573 CGSB38 16748274 IC50 = 20 nM T86573 CIC18J 16748525 IC50 = 29 nM T86573 CD57VL 16748526 IC50 = 20 nM T86573 CUQG95 16748527 IC50 = 10 nM T86573 CN1P8T 16748528 IC50 = 17 nM T86573 CYWJ25 16748529 IC50 = 22 nM T86573 CY64OX 16748634 IC50 = 59 nM T86573 CCTY21 16748636 IC50 = 431 nM T86573 C1DU6C 16748637 IC50 = 53 nM T86573 CH5E8D 16748745 IC50 = 11 nM T86573 CT8S1K 17032699 IC50 > 5000 nM T86573 CQT58O 17033137 IC50 > 5000 nM T86573 CS1LN8 17033372 IC50 > 5000 nM T86573 CSU17Z 18184806 IC50 = 400 nM T86573 CUWA47 18467513 IC50 = 380 nM T86573 C3LSH2 19165245 IC50 >= 5000 nM T86573 CZUJ07 19168353 IC50 >= 5000 nM T86573 C7ZL3T 19168356 IC50 >= 5000 nM T86573 CB62FV 20766912 IC50 > 10000 nM T86573 CVR34M 20766928 IC50 > 5000 nM T86573 CTMK79 20766951 IC50 > 10000 nM T86573 CEW1H6 20766964 IC50 > 10000 nM T86573 CF6VY0 21343422 IC50 = 28 nM T86573 CMFZ98 21343423 IC50 = 47 nM T86573 CKBR14 21343449 IC50 = 45 nM T86573 CR8PG0 22058483 IC50 = 200 nM T86573 CJEA25 22058485 IC50 = 170 nM T86573 C82WXQ 22058487 IC50 = 130 nM T86573 CMW8Z1 22058491 IC50 = 74 nM T86573 C9RN7Y 22058493 IC50 = 18 nM T86573 CDN25T 22058495 IC50 = 890 nM T86573 CW59LM 22058498 IC50 = 66 nM T86573 C0N5HJ 22058499 IC50 = 300 nM T86573 CG1ET0 22058500 IC50 = 210 nM T86573 C80VAD 22058504 IC50 > 10000 nM T86573 C50PZT 22058514 IC50 = 630 nM T86573 C2XKA3 22058516 IC50 = 540 nM T86573 CHD96V 22058517 IC50 = 140 nM T86573 CZQ9S0 22058521 IC50 = 260 nM T86573 C1SQF5 22058523 IC50 = 210 nM T86573 CG1XV3 22058530 IC50 = 35 nM T86573 C8QYM5 22058533 IC50 = 110 nM T86573 CFY48L 22058535 IC50 = 130 nM T86573 C98PNG 22058536 IC50 = 870 nM T86573 CQV4C5 22058537 IC50 = 210 nM T86573 CT81BG 22058540 IC50 = 330 nM T86573 C50SZG 22058546 IC50 = 230 nM T86573 CJ0E2N 22058549 IC50 = 410 nM T86573 CUV9T5 22058554 IC50 = 120 nM T86573 CN61PF 22058555 IC50 = 60 nM T86573 C05UQA 22093099 IC50 = 180 nM T86573 CVA2J7 22093112 IC50 = 110 nM T86573 CIEV83 22226545 IC50 > 5000 nM T86573 CO5D4T 22238480 IC50 = 64 nM T86573 C8NFO7 22238485 IC50 = 230 nM T86573 C8Z7YO 22238488 IC50 = 360 nM T86573 C8Z7TF 22238492 IC50 = 130 nM T86573 C4RL8K 22238495 IC50 = 220 nM T86573 CHD0W4 22238496 IC50 = 500 nM T86573 CS4O3X 22349495 IC50 > 1000 nM T86573 C2J8FN 22349571 IC50 = 160 nM T86573 C2E5SM 22459608 IC50 = 41 nM T86573 CF2W6L 22459610 IC50 = 120 nM T86573 C0AF6L 22459619 IC50 = 44 nM T86573 CYBK83 22459624 IC50 = 170 nM T86573 C5BEX9 22459627 IC50 = 110 nM T86573 CP21KX 22459655 IC50 = 190 nM T86573 CMO17X 22459661 IC50 = 410 nM T86573 CG68HF 22459673 IC50 = 54 nM T86573 CDB6I3 22459677 IC50 = 310 nM T86573 C38PCH 22459686 IC50 = 76 nM T86573 C9O4YG 22459693 IC50 = 760 nM T86573 C6PF0W 22459706 IC50 = 32 nM T86573 CK1W8G 22459707 IC50 > 1600 nM T86573 C65GMW 22459716 IC50 = 78 nM T86573 CEJ85U 22459723 IC50 > 5000 nM T86573 CTIL79 22459725 IC50 = 160 nM T86573 C2R1IB 22459727 IC50 = 300 nM T86573 C97UNB 22459730 IC50 = 410 nM T86573 CLK5B2 22459738 IC50 = 330 nM T86573 CSQ68W 22459746 IC50 = 100 nM T86573 C0E7BC 22459748 IC50 = 59 nM T86573 C7BNW0 22459765 IC50 = 130 nM T86573 CIT2G5 22459770 IC50 = 330 nM T86573 C4RI2U 22459775 IC50 > 10000 nM T86573 C5PST6 22459779 IC50 = 41 nM T86573 C0CYK4 22459787 IC50 = 21 nM T86573 CIK04R 22558406 IC50 > 10000 nM T86573 C63IGS 22946285 IC50 = 640 nM T86573 CMF8R1 22946293 IC50 = 43 nM T86573 CS42ZC 23626089 IC50 = 4100 nM T86573 CJO79M 23644735 Ki = 255 nM T86573 C2NW5X 23648220 Ki = 84 nM T86573 CCN63I 23648221 Ki = 143 nM T86573 CMVH63 23648222 Ki = 27 nM T86573 C0OR1M 23648223 Ki = 153 nM T86573 C5PIF4 23648224 Ki = 169 nM T86573 C90FQM 23648225 Ki = 49 nM T86573 CB35PV 23648226 Ki = 94 nM T86573 CQ90NK 23648227 Ki = 14 nM T86573 CKZT87 23648228 Ki = 108 nM T86573 CBC71W 23648229 Ki = 38 nM T86573 CH3Z4Q 24513583 IC50 > 5000 nM T86573 CBU17V 24513606 IC50 > 5000 nM T86573 CDXA20 24513641 IC50 > 5000 nM T86573 CZ8MT3 24517453 IC50 > 5000 nM T86573 CU94DR 24538043 IC50 > 5000 nM T86573 CYG18K 24748985 Ki = 540 nM T86573 C6M4QN 24748986 Ki = 1700 nM T86573 CK32AR 24749071 Ki = 1100 nM T86573 C9E0AU 24749072 Ki = 650 nM T86573 CG3O4V 24999500 IC50 > 5000 nM T86573 CO6DB0 25147739 Ki = 170 nM T86573 C09KIE 25181866 Ki = 1200 nM T86573 CND10S 25181867 Ki = 11000 nM T86573 CX5BU0 25181868 Ki = 340 nM T86573 C68PMG 25181869 Ki = 2600 nM T86573 C5JVN4 25210968 Ki = 8700 nM T86573 CUZT43 25210969 Ki = 2300 nM T86573 CW8I0P 25879063 IC50 = 87.7 nM T86573 CFU76P 26196040 IC50 = 1790 nM T86573 CS23HG 44024165 IC50 > 5000 nM T86573 C5IL9F 44024167 IC50 > 5000 nM T86573 C0F8KP 44275519 IC50 = 50 nM T86573 CQ2I6J 44275642 IC50 > 10000 nM T86573 C5YN8D 44275688 IC50 = 30 nM T86573 CQ4E9F 44275711 IC50 > 10000 nM T86573 CY8L1G 44275942 IC50 > 10000 nM T86573 CE0HC9 44276467 IC50 = 18 nM T86573 CEH64S 44276468 IC50 = 3800 nM T86573 C24IPY 44276469 IC50 = 740 nM T86573 C3DW1Z 44276622 IC50 = 550 nM T86573 C9YKC1 44276665 IC50 = 60 nM T86573 C4RZE0 44276698 IC50 = 820 nM T86573 CML9P3 44276709 IC50 = 3000 nM T86573 C1BZ8S 44276733 IC50 = 1660 nM T86573 C2BCQ0 44276734 IC50 = 740 nM T86573 CALV53 44276798 IC50 > 5000 nM T86573 CDB20G 44276803 IC50 > 5000 nM T86573 CZ2X8G 44276804 IC50 > 5000 nM T86573 C5GJ8H 44276818 IC50 > 1700 nM T86573 CD87HW 44276819 IC50 > 5000 nM T86573 CF18UY 44276869 IC50 = 150 nM T86573 C37KLD 44276961 IC50 = 400 nM T86573 C7TYB8 44276962 IC50 = 247 nM T86573 CT2Q0G 44276963 IC50 > 5000 nM T86573 CH3PF8 44277008 IC50 > 5000 nM T86573 CDS04H 44277009 IC50 = 1200 nM T86573 CIYN69 44304863 IC50 = 500 nM T86573 C0VD6L 44304866 IC50 > 5000 nM T86573 CS9FU7 44304883 IC50 = 41 nM T86573 CO3VX9 44304884 IC50 = 91 nM T86573 C50RLI 44304885 IC50 > 5000 nM T86573 CYF62T 44304900 IC50 > 5000 nM T86573 C84LXP 44304912 IC50 = 310 nM T86573 CH3UY4 44304932 IC50 = 100 nM T86573 CFG8V3 44305013 IC50 = 21 nM T86573 CSH83K 44305029 IC50 > 2000 nM T86573 CH6U5M 44305031 IC50 > 5000 nM T86573 CL60QO 44305034 IC50 > 1600 nM T86573 C0ZV6T 44305048 IC50 > 5000 nM T86573 C95JXK 44305067 IC50 = 1600 nM T86573 CNZ9E0 44305078 IC50 > 5000 nM T86573 CA3PV5 44305083 IC50 = 88 nM T86573 C94HVX 44305086 IC50 = 190 nM T86573 C7HFJ9 44305087 IC50 = 210 nM T86573 CNFR41 44305128 IC50 > 340 nM T86573 C27MSW 44305145 IC50 > 5000 nM T86573 CRQC38 44305148 IC50 > 57 nM T86573 CB40FT 44305192 IC50 > 5000 nM T86573 CKV9A4 44305213 IC50 > 2000 nM T86573 C7KEI3 44305214 IC50 > 2000 nM T86573 CGLZ25 44305233 IC50 > 5000 nM T86573 C5KRW0 44307938 IC50 = 72 nM T86573 CO0YU5 44308038 IC50 = 270 nM T86573 C3SEZ1 44308050 IC50 = 78 nM T86573 CGBD53 44308081 IC50 = 290 nM T86573 C2TN9P 44308105 IC50 = 3500 nM T86573 CAOH09 44308165 IC50 = 720 nM T86573 CYP86T 44308220 IC50 = 130 nM T86573 CKSV35 44308227 IC50 > 1000 nM T86573 CKSW94 44308417 IC50 = 250 nM T86573 CMP04J 44308425 IC50 = 620 nM T86573 CY2J8B 44329217 IC50 = 75 nM T86573 CLVU19 44329328 IC50 = 57 nM T86573 CQ1MW8 44329361 IC50 = 630 nM T86573 C2SG3Z 44329366 IC50 = 590 nM T86573 CRV1W0 44329410 IC50 > 3000 nM T86573 CFJ8S1 44329515 IC50 = 960 nM T86573 C7UX0J 44329529 IC50 = 110 nM T86573 C8GJN2 44329556 IC50 = 630 nM T86573 CA8P2J 44329800 IC50 > 1000 nM T86573 CPS1I4 44329801 IC50 = 2500 nM T86573 CMZ1T2 44329808 IC50 = 810 nM T86573 CF8P9E 44329815 IC50 > 1000 nM T86573 C50YRM 44330611 IC50 = 330 nM T86573 CZ2BR4 44330738 IC50 > 3000 nM T86573 C2N5CJ 44330750 IC50 = 130 nM T86573 CZ9UE0 44330773 IC50 = 340 nM T86573 CW8LY7 44330809 IC50 = 660 nM T86573 C07CSW 44330826 IC50 > 3000 nM T86573 CG17NB 44330827 IC50 = 240 nM T86573 CBN9J6 44330828 IC50 = 340 nM T86573 CB1VJ4 44336201 IC50 = 110 nM T86573 C4J8MO 44340409 IC50 = 40 nM T86573 C8BTY0 44340410 IC50 = 11 nM T86573 CL3OG8 44340423 IC50 = 200 nM T86573 C5FE6B 44340424 IC50 = 35 nM T86573 COW8S4 44340430 IC50 = 205 nM T86573 CQ4S0B 44340431 IC50 = 38 nM T86573 C9GB2W 44340450 IC50 > 5000 nM T86573 CLXS31 44340666 IC50 = 93 nM T86573 CU5N8R 44340674 IC50 > 5000 nM T86573 CX5HD2 44340724 IC50 = 35 nM T86573 CQC6A8 44340732 IC50 = 77 nM T86573 CRV2S9 44345136 IC50 = 84 nM T86573 CW4D9K 44345137 IC50 = 266 nM T86573 CHX1C3 44345138 IC50 = 6 nM T86573 CHJ67K 44345267 IC50 = 290 nM T86573 CQ52KT 44345310 IC50 = 420 nM T86573 C1AN9S 44345333 IC50 = 260 nM T86573 CTO57X 44354730 IC50 > 100000 nM T86573 CJ3N4G 44354906 IC50 = 89.8 nM T86573 CX9C7V 44355016 IC50 = 975 nM T86573 C4I3GD 44367217 IC50 = 160 nM T86573 CE9OC4 44367244 IC50 = 19 nM T86573 CB41DS 44367248 IC50 = 43 nM T86573 C5X1GF 44367255 IC50 = 46 nM T86573 C91HWG 44367420 IC50 = 26 nM T86573 CG45ZL 44367512 IC50 = 83 nM T86573 CU1VX2 44367513 IC50 < 10 nM T86573 C0RXO6 44367526 IC50 = 65 nM T86573 CXM9L0 44367538 IC50 = 5 nM T86573 CWIO57 44367546 IC50 = 180 nM T86573 CRE48F 44367552 IC50 = 65 nM T86573 CJR86I 44367578 IC50 = 29 nM T86573 CZID50 44367579 IC50 < 5 nM T86573 CY0OA1 44367590 IC50 > 10000 nM T86573 CZSP50 44367614 IC50 = 43 nM T86573 CZYC59 44367615 IC50 = 5 nM T86573 CY2J7R 44367639 IC50 = 30 nM T86573 CT5DZ1 44367690 IC50 = 21 nM T86573 COXS41 44367703 IC50 < 50 nM T86573 CS45OJ 44367718 IC50 = 33 nM T86573 CZU5N0 44367719 IC50 = 21 nM T86573 C4SOR5 44367730 IC50 = 5 nM T86573 C6VAS4 44367731 IC50 = 53 nM T86573 CM9S8K 44367733 IC50 = 140 nM T86573 CM06LV 44367743 IC50 = 15 nM T86573 CJ98VU 44367747 IC50 = 15 nM T86573 CR65TE 44390711 IC50 = 30 nM T86573 CSX2D6 44390718 IC50 = 17 nM T86573 C34JFM 44390721 IC50 = 91 nM T86573 CUY3T1 44390765 IC50 = 47 nM T86573 C1SNV9 44390777 IC50 = 22 nM T86573 CFI5P2 44390789 IC50 = 1710 nM T86573 CBQ8I7 44390790 IC50 = 100 nM T86573 C4P1JT 44390791 IC50 = 297 nM T86573 C8RDA1 44390811 IC50 = 821 nM T86573 C5B2FZ 44390828 IC50 = 71 nM T86573 CPZ9H5 44405422 IC50 = 192 nM T86573 C5LNB2 44405423 IC50 = 94 nM T86573 CN3O2U 44405428 IC50 = 49 nM T86573 C4FC9Y 44405429 IC50 = 328 nM T86573 CL0AE9 44405441 IC50 = 526 nM T86573 CNKD60 44405446 IC50 = 96 nM T86573 CK3PY1 44405447 IC50 = 104 nM T86573 C3R6PV 44405453 IC50 = 80 nM T86573 C7ZP0M 44405472 IC50 = 51 nM T86573 CZR84O 44405475 IC50 = 45 nM T86573 CY5N0I 44405476 IC50 = 68 nM T86573 CM0OF7 44405514 IC50 = 119 nM T86573 CH53NE 44405515 IC50 = 393 nM T86573 CR2Z7O 44405520 IC50 = 64 nM T86573 CG43TN 44405539 IC50 = 369 nM T86573 C5MA9V 44405578 IC50 = 71 nM T86573 CES5D6 44405580 IC50 = 79 nM T86573 CB43CW 44405581 IC50 = 948 nM T86573 CLG35S 44410469 IC50 = 71800 nM T86573 C3JM4T 44410476 IC50 = 222 nM T86573 CRP9B7 44410594 IC50 = 17000 nM T86573 CNE08X 44410595 IC50 = 1170 nM T86573 C0G5WM 44410601 IC50 = 128 nM T86573 C5R1BT 44410602 IC50 = 19500 nM T86573 C3SZT7 44410608 IC50 = 1360 nM T86573 COY6D8 44410643 IC50 = 4040 nM T86573 C8L3EA 44410644 IC50 = 7680 nM T86573 C6CS4Y 44410726 IC50 = 21000 nM T86573 C8ZP5U 44410728 IC50 = 7850 nM T86573 CO6K7B 44410732 IC50 = 58400 nM T86573 C8H4ES 44410734 IC50 = 6210 nM T86573 C48CJL 44410735 IC50 = 364 nM T86573 CJ81XI 44410872 IC50 = 27900 nM T86573 CMAZ04 44412558 IC50 = 246 nM T86573 CFQA81 44412573 IC50 > 1000 nM T86573 CL8JF5 44412582 IC50 = 273 nM T86573 C4PO0Y 44412597 IC50 = 96 nM T86573 CR61JY 44412598 IC50 = 86 nM T86573 CW4YP0 44412618 IC50 = 506 nM T86573 C4P8QV 44412632 IC50 = 68 nM T86573 C4Y6EC 44412633 IC50 = 24 nM T86573 CP0LU8 44412648 IC50 = 132 nM T86573 C1UP8I 44412712 IC50 = 93 nM T86573 C95XHE 44412713 IC50 > 1000 nM T86573 CFP3B7 44412731 IC50 > 1000 nM T86573 CR4N1Y 44412759 IC50 = 499 nM T86573 C5EP3N 44412773 IC50 = 785 nM T86573 C8LRG7 44412774 IC50 = 749 nM T86573 CAQC52 44412793 IC50 = 498 nM T86573 C70YFO 44415246 Ki = 60 nM T86573 CRZW96 44415248 Ki = 37 nM T86573 C16EMS 44433349 IC50 = 72000 nM T86573 CC2UO4 44440695 IC50 = 18800 nM T86573 CY6SQ1 44458844 IC50 = 150 nM T86573 C0RU5A 44458846 IC50 = 290 nM T86573 C14SVM 44458898 IC50 > 1000 nM T86573 COQ83H 44578784 IC50 = 18800 nM T86573 C84EYU 44578785 Ki = 310 nM T86573 C8GJB9 44578786 Ki = 180 nM T86573 C9T2EI 44578787 Ki = 440 nM T86573 CIK76G 44578789 Ki > 100000 nM T86573 CEI32X 44589747 Ki = 14300 nM T86573 C2MF0S 44589785 Ki > 100000 nM T86573 CG7WJ4 44589786 Ki = 30100 nM T86573 C7Y9QT 44602364 IC50 > 5000 nM T86573 CM2U4H 45257259 IC50 > 5000 nM T86573 CAH41O 45257352 IC50 > 5000 nM T86573 C7OGF2 45257354 IC50 > 5000 nM T86573 CVO20H 46839190 Ki = 2200 nM T86573 C3GET9 46839191 Ki = 34 nM T86573 C0SV8O 46839192 Ki = 200 nM T86573 C1V3CQ 46839320 Ki = 44 nM T86573 CH6S4E 46871958 IC50 > 5000 nM T86573 CG2JO0 46876259 Ki = 300 nM T86573 C01DSF 46876831 Ki = 950 nM T86573 CG3RM9 46876832 Ki = 290 nM T86573 CJQ8D6 46898106 IC50 > 5000 nM T86573 CIT31Y 46927861 Ki = 250 nM T86573 CXW02B 46927862 Ki = 120 nM T86573 CU4Z3R 49864088 Ki = 1400 nM T86573 CP5HR1 49864089 Ki = 1500 nM T86573 CQ39WM 49864090 Ki = 230 nM T86573 C76JYP 49864102 Ki = 1200 nM T86573 CN2G3Z 49864103 Ki = 1800 nM T86573 C01GAC 49864104 Ki = 200 nM T86573 CR8E0Z 51351534 Ki = 24 nM T86573 C9YL2W 51351535 Ki = 73 nM T86573 CPY1M0 51351558 Ki = 38 nM T86573 C09MCD 52589406 IC50 > 5000 nM T86573 CT64YQ 52905544 Ki = 487 nM T86573 C81NCO 53317433 Ki = 770 nM T86573 C81TOB 53317434 Ki = 167 nM T86573 C7R4DT 53317435 Ki = 83 nM T86573 CZ4FR9 53317436 Ki = 34 nM T86573 C0MC6P 53320028 Ki = 3770 nM T86573 C64FAH 53320029 Ki = 6600 nM T86573 CQU37F 53320030 Ki = 39 nM T86573 CFO5E7 53320031 Ki = 44 nM T86573 CN32LO 53320311 Ki = 84 nM T86573 CPO0F3 53322659 Ki = 60 nM T86573 CMT39Y 53322660 Ki = 1900 nM T86573 CN6Q8M 53324226 Ki = 14 nM T86573 CC9D8J 53326788 Ki = 30 nM T86573 C6HQ7S 56835081 IC50 = 2100 nM T86573 C18UZI 56835082 IC50 = 4500 nM T86573 C91ARE 56835083 IC50 = 8800 nM T86573 CNGX19 56835085 IC50 = 3200 nM T86573 C5HZ3Q 56835102 IC50 = 2800 nM T86573 CP32QL 57391310 IC50 > 5000 nM T86573 CBMX91 57391311 IC50 > 5000 nM T86573 CCZ98A 57393086 IC50 > 5000 nM T86573 CK1RZ4 57394813 IC50 > 5000 nM T86573 C5BNH7 57396578 IC50 > 5000 nM T86573 C3HKO1 57398354 IC50 > 5000 nM T86573 CMAT05 57398355 IC50 > 5000 nM T86573 CM7T2I 57398356 IC50 > 5000 nM T86573 C6V0XL 57398357 IC50 > 5000 nM T86573 C3XD9L 57400014 IC50 > 5000 nM T86573 CR6AE3 57400851 IC50 = 400 nM T86573 C7HF5T 57401823 IC50 > 5000 nM T86573 C4IE8C 57401824 IC50 > 5000 nM T86573 CY5L8X 57401825 IC50 > 5000 nM T86573 CF79PO 57403530 IC50 > 5000 nM T86573 CC54BA 57403531 IC50 > 5000 nM T86573 C09ZCY 59053796 IC50 = 28860 nM T86573 C48TLR 59053798 IC50 = 73240 nM T86573 CB9G6K 67473072 IC50 >= 5000 nM T86573 C4DG7M 67473106 IC50 > 5000 nM T86573 CHW41M 67473122 IC50 >= 5000 nM T86573 C87ORP 67473132 IC50 >= 5000 nM T86573 CEU7I8 67473135 IC50 >= 5000 nM T86573 C3WLG5 67473139 IC50 >= 5000 nM T86573 CO5U4S 70693788 IC50 = 6430 nM T86573 C3IQE9 70850880 IC50 > 5000 nM T86573 CH26JV 70851038 IC50 > 5000 nM T86573 CF53JE 71297189 IC50 > 5000 nM T86573 CFA3N8 71450059 IC50 >= 5000 nM T86573 CMI97N 71453700 IC50 >= 5000 nM T86573 CW3VL9 71453701 IC50 >= 5000 nM T86573 CM05XU 71455424 IC50 >= 5000 nM T86573 C61ATW 71455425 IC50 >= 5000 nM T86573 C3AT8D 71462576 IC50 >= 5000 nM T86573 CZAV85 71462577 IC50 >= 5000 nM T86573 CMVL76 71661540 IC50 > 5000 nM T86573 C1V5AQ 71661543 IC50 > 5000 nM T86573 CX5WE1 71661544 IC50 > 5000 nM T86573 CV1D5W 71661721 IC50 > 5000 nM T86573 CNIJ92 71661722 IC50 > 5000 nM T86573 CO36TX 71661724 IC50 > 5000 nM T86573 CZ1TF2 71661725 IC50 > 5000 nM T86573 CW54QI 71661894 Ki > 5000 nM T86573 CC9U7A 71661895 IC50 > 5000 nM T86573 C8CX0T 71661896 IC50 > 5000 nM T86573 C6RN9G 71661897 IC50 > 5000 nM T86573 CI6YS9 71662079 IC50 > 5000 nM T86573 C87LXA 71662080 IC50 > 5000 nM T86573 C51OLK 71662081 Ki > 5000 nM T86573 C2ILR9 71662082 IC50 > 5000 nM T86573 C7IQA2 71662258 IC50 > 5000 nM T86573 CD35JI 71662259 IC50 > 5000 nM T86573 CIFH53 71662260 IC50 > 5000 nM T86573 CRB19S 71662261 IC50 > 5000 nM T86573 CP6WC3 71662422 IC50 > 5000 nM T86573 C6T5XE 71662423 IC50 > 5000 nM T86573 CE0ON2 71662424 IC50 > 5000 nM T86573 CD9UX5 71662426 IC50 > 5000 nM T86573 CYT20K 71662586 IC50 > 5000 nM T86573 CO8V4B 71662587 IC50 > 5000 nM T86573 CC0A9E 71662588 IC50 > 5000 nM T86573 C50TWZ 71662589 IC50 > 5000 nM T86573 C9GAL6 71662590 IC50 > 5000 nM T86573 CX58GA 71662775 Ki > 5000 nM T86573 C8N7CG 71662776 IC50 > 5000 nM T86573 CC3WB6 71662779 IC50 > 5000 nM T86573 CDVK12 71662780 IC50 > 5000 nM T86573 C39KQY 71716568 IC50 = 90 nM T86573 C3M0JK 72163956 IC50 = 98 nM T86573 CNQ2D6 72945146 Ki = 165 nM T86573 C5OJ0X 72945148 Ki = 186 nM T86573 C01HVL 72945149 Ki = 102 nM T86573 C1OVC0 72945150 Ki = 231 nM T86573 CBPC50 72945349 Ki = 84 nM T86573 C7MJQ5 72945350 Ki = 967 nM T86573 C9NTH1 72945351 Ki = 175 nM T86573 CVJ0N8 72945352 Ki = 70 nM T86573 CP1I9N 72945353 Ki = 1964 nM T86573 CJ4R8C 72945541 Ki = 1227 nM T86573 C74WCI 72945542 Ki = 88 nM T86573 C7T3HN 72945732 Ki = 24 nM T86573 C95BZQ 72947911 Ki = 15 nM T86573 CCVO01 72947912 Ki = 14 nM T86573 CB7HG8 72948102 Ki = 37 nM T86573 C4U3OA 72948103 Ki = 56 nM T86573 CX2U3L 72948104 Ki = 44 nM T86573 C3N7OD 72948105 Ki = 749 nM T86573 CZJ5F6 73346517 Ki = 2398 nM T86573 CN5QE0 73346518 Ki = 321 nM T86573 C26EXZ 73349141 IC50 = 330 nM T86573 CAD90T 73349545 Ki = 437 nM T86573 CD4BY1 73351103 Ki = 2672 nM T86573 CB94EM 73352218 IC50 = 387 nM T86573 CWO9Q0 73352572 Ki = 163 nM T86573 CPS4I8 76309998 Ki = 12.6 nM T86573 CB2PT6 76309999 Ki = 40 nM T86573 CL42ER 76310000 Ki = 215 nM T86573 CI1J4W 76310001 Ki = 94 nM T86573 CEB47C 76310002 Ki = 2790 nM T86573 C3ICR7 76310003 Ki = 524 nM T86573 C7C9FJ 76317234 Ki = 235 nM T86573 CTLJ38 76317235 Ki = 364 nM T86573 CZ9U2T 76320941 Ki = 233 nM T86573 C7HJC1 76324606 Ki = 188 nM T86573 C0DFQ1 76328163 Ki = 438 nM T86573 CL41TU 76328164 Ki = 134 nM T86573 C86TRQ 76331843 Ki = 174 nM T86573 CTFG08 76331844 Ki = 147 nM T86573 C3OVW6 76335415 Ki = 188 nM T86573 CG7Z4S 76335416 Ki = 188 nM T86573 C72ZFE 90663687 IC50 = 800 nM T86573 CD9S8B 90663694 Ki = 110 nM T86573 CC6RG7 90663712 IC50 = 175000 nM T86573 CEX1D3 90663714 IC50 = 800 nM T86573 C0A3ZW 90663715 IC50 = 6000 nM T86573 C47LAF 135418940 IC50 > 10000 nM T86573 CJVW76 135419254 IC50 = 52800 nM T86573 C8J2PC 135456762 IC50 > 10000 nM T86573 CEDB45 135500033 IC50 = 18 nM T86573 C4BFY3 135566969 IC50 > 10000 nM T86573 C0USX4 135883678 IC50 = 740 nM T86573 CM9QB3 135883679 IC50 = 800 nM T86573 C3GW8I 135883680 IC50 > 1000 nM T86573 CIT3E5 135976449 IC50 = 37000 nM T86573 C25EPJ 135976460 IC50 > 1000000 nM T86573 CMG6I4 135976469 IC50 = 440 nM T86573 CV4G0A 135976470 IC50 > 1000000 nM T86573 CQ4T2N 135976471 IC50 = 132000 nM T86573 CF0GR8 135976472 IC50 > 1000000 nM T86573 CTZ82I 135976473 IC50 = 1200 nM T86573 CV9WK5 135976474 IC50 = 1000 nM T86573 C5W3TV 135976476 IC50 = 1320 nM T86573 C0UR9J 135976481 IC50 = 460000 nM T86573 CTF7A4 136042356 IC50 > 5000 nM T86573 CY94ZB 136215772 IC50 > 10000 nM T86573 C7JEG1 136215773 IC50 > 10000 nM T86573 CF7O2U 136215774 IC50 > 10000 nM T86573 CFP0V5 136215897 IC50 > 10000 nM T86573 C3NHA6 136219159 IC50 > 5000 nM T86573 CG75EV 138393087 Ki > 5000 nM T86573 C1GPY5 145952889 IC50 = 1500 nM T86573 CFQ2O9 145954131 IC50 > 30000 nM T86573 C8O2IJ 145963797 Ki > 5000 nM T86573 C40WKT 145964095 Ki > 5000 nM T86573 CR78JK 145964212 Ki > 5000 nM T86573 CFS5Z3 145964258 Ki > 5000 nM T86573 CC3T5V 145964499 Ki > 5000 nM T86573 C0KGT4 145964791 Ki > 5000 nM T86573 CJAI17 145964939 Ki > 5000 nM T86573 C3AXP6 145965235 Ki > 5000 nM T86573 CW50CM 145965999 Ki > 5000 nM T86573 CB4NX2 145966576 Ki > 5000 nM T86573 C5V7ZK 145966629 Ki > 5000 nM T86573 C8E7TL 145966683 Ki > 5000 nM T86573 C02DKL 145966779 Ki > 5000 nM T86573 C5K3DS 145967011 Ki > 5000 nM T86573 C1AD8R 145967013 Ki > 5000 nM T86573 CYTB64 145967134 Ki > 5000 nM T86573 C9EZ5L 145970298 Ki > 5000 nM T86573 C4RNH8 145970986 Ki = 2900 nM T86573 C5GW7N 145971015 Ki > 5000 nM T86573 CA6C2F 145972082 Ki > 5000 nM T86573 C2PV6E 145972358 Ki > 5000 nM T86573 CTV68U 145972501 Ki > 5000 nM T86573 C5HCJ8 145972590 Ki > 5000 nM T86573 CI31YE 145972757 IC50 = 4540 nM T86573 CFS82G 145973482 Ki > 5000 nM T86573 C06FRK 145974169 Ki > 5000 nM T86573 C1KSO5 145974525 Ki = 3300 nM T86573 C8B7LI 145974642 Ki > 5000 nM T86573 C24ZLQ 145974896 Ki > 5000 nM T86573 C1VID9 145975055 Ki > 5000 nM T86573 C7RUP4 145975474 Ki > 5000 nM T86573 C23DWC 145975793 Ki > 5000 nM T86573 CR1ND4 145975885 Ki > 5000 nM T86573 C3ZQ7I 145976477 Ki = 2000 nM T86573 C48WSM 145976500 Ki > 5000 nM T86573 CHA9M2 145976564 Ki > 5000 nM T86573 C1KJ4W 145977312 Ki > 5000 nM T86573 CC1L4J 145977399 Ki > 5000 nM T86573 C2GU3O 145977423 Ki > 5000 nM T86573 CG86KY 145977474 Ki > 5000 nM T86573 CTGB02 145977680 Ki > 5000 nM T86573 CJX17G 145977828 Ki = 2300 nM T86573 CZK4L8 145978048 Ki > 5000 nM T86573 CQF9Z2 145978149 Ki > 5000 nM T86573 C06RKZ 145978312 Ki > 5000 nM T86573 C24OSG 145979776 IC50 = 7380 nM T86573 C93AKF 145980356 IC50 = 1600 nM T86573 C67YXK 145980711 IC50 = 4200 nM T86573 CUSP05 145981621 IC50 = 360 nM T86573 C10YDI 145982128 IC50 = 430 nM T86573 CWC78S 145983656 IC50 = 1200 nM T86573 C6VP2S 145985880 IC50 > 30000 nM T86573 CPLR18 145988080 IC50 = 570 nM T86573 C1K4BC 145989436 IC50 = 360 nM T86573 C5QBJ2 145989469 IC50 = 4400 nM T86573 CCY78M 145990077 IC50 = 660 nM T86573 C20PUW 145990385 IC50 = 2200 nM T86573 CIG96S 145990435 IC50 = 790 nM T86573 CBL59V 145990969 IC50 = 4500 nM T86573 CP42FJ 145991406 IC50 = 1200 nM T86573 D01LDQ 24749070 Ki = 30 nM T86573 D02YMQ 44410733 IC50 = 456 nM T86573 D03HDS 6475540 Ki = 380 nM T86573 D04LRN 22238481 IC50 = 600 nM T86573 D05SKE 44410796 IC50 = 408 nM T86573 D06FSR 2307681 IC50 = 7660 nM T86573 D06RQV 44410708 IC50 = 419 nM T86573 D07BPT 135457978 IC50 > 10000 nM T86573 D07HZQ 444451 Ki = 21 nM T86573 D08OSM 10607518 IC50 = 5840 nM T86573 D0A0UW 22238483 IC50 = 500 nM T86573 D0A4AL 477579 Ki = 250 nM T86573 D0AL2E 44410707 IC50 = 524 nM T86573 D0B2WX 135407310 IC50 > 10000 nM T86573 D0D1KZ 87894 IC50 = 6840 nM T86573 D0D2ST 11962095 IC50 = 343 nM T86573 D0E5EW 135531482 IC50 > 10000 nM T86573 D0G3BY 44410465 IC50 = 15400 nM T86573 D0GA0Y 135463623 IC50 > 10000 nM T86573 D0H1II 510913 IC50 = 630 nM T86573 D0J9OS 44410800 IC50 = 6210 nM T86573 D0K4EM 44410928 IC50 = 637 nM T86573 D0L0MJ 644354 IC50 = 1150 nM T86573 D0L0ZP 15462732 IC50 = 8200 nM T86573 D0Q3WC 44410473 IC50 = 1110 nM T86573 D0S4BK 73680 Ki = 100 nM T86573 D0T4UE 44578788 Ki = 4000 nM T86573 D0V0YP 44410875 IC50 = 2320 nM T86573 D0Y1MH 135471354 IC50 > 10000 nM T86573 D0Z0YB 16748635 IC50 = 2200 nM T86573 D0Z8EV 446541 Ki = 6 nM T86573 D0ZG3O 44410730 IC50 = 586 nM T40890 D0R9YR 64971 IC50 = 32000 nM T40890 C8NW5J 3815 IC50 = 1800 nM T40890 CZP38H 161352 IC50 > 200000 nM T40890 CS5B8N 421610 IC50 = 40000 nM T40890 C1D0RN 5470187 IC50 = 7100 nM T40890 C6B5HR 5482346 IC50 = 1800 nM T40890 CGFB94 11232674 IC50 = 1800 nM T40890 CHS62D 11268312 IC50 = 1800 nM T40890 C3KGN1 11613161 IC50 = 620 nM T40890 CAP7Q3 12305768 IC50 = 42000 nM T40890 CSL5K8 21672700 IC50 = 38000 nM T40890 CH6W7F 44189870 IC50 = 9400 nM T40890 C5BH9A 44190064 IC50 = 11400 nM T40890 CON09V 44190252 IC50 = 6900 nM T40890 CCI7E3 44588609 IC50 = 133000 nM T40890 CZ8V3H 45268743 IC50 = 11400 nM T40890 CU2S0Y 46898040 IC50 = 2600 nM T40890 C7N3CS 46898044 IC50 = 1600 nM T40890 CU25CB 49864133 IC50 = 660 nM T40890 CI5M9E 68911124 IC50 = 30000 nM T40890 C3H0XF 91184682 IC50 = 10000 nM T40890 CD61RK 102142142 IC50 = 15850 nM T40890 CR0H7N 102142143 IC50 = 12530 nM T40890 CT45VC 145964783 IC50 > 25000 nM T40890 CY6CS5 145965005 IC50 > 25000 nM T40890 C0BFD4 145965512 IC50 > 25000 nM T40890 CXA3T5 145965880 IC50 > 25000 nM T40890 CY89HE 145970487 IC50 = 8980 nM T40890 C15XCS 145971009 IC50 > 25000 nM T40890 CB4VN1 145971626 IC50 > 25000 nM T40890 CL8O4C 145971811 IC50 = 740 nM T40890 C0QKI8 145972528 IC50 > 25000 nM T40890 CGN3T0 145973063 IC50 > 25000 nM T40890 CV5DG9 145973331 IC50 = 12340 nM T40890 CZX46S 145976815 IC50 > 25000 nM T40890 C3V2QY 145977921 IC50 > 25000 nM T40890 CW4P8G 145978332 IC50 = 5380 nM T40890 CXAK63 145978784 IC50 = 640 nM T40890 D05UKJ 442972 IC50 = 5000 nM T60529 D00IBN 54676228 IC50 = 1300 nM T60529 D03RTS 2662 IC50 = 50 nM T60529 D04YMH 151166 IC50 = 7 nM T60529 D05FTJ 4044 IC50 = 25000 nM T60529 D05VLS 5090 IC50 = 1900 nM T60529 D06YPU 39912 IC50 = 98.65 nM T60529 D07BPS 5359 IC50 = 560 nM T60529 D07HBX 338 IC50 = 500000 nM T60529 D07UYO 441401 IC50 = 8190 nM T60529 D08IFL 4037 IC50 = 220 nM T60529 D09JUG 60490 IC50 > 10000 nM T60529 D09MGR 123619 IC50 = 98800 nM T60529 D0A1PX 3394 IC50 = 10 nM T60529 D0B2WJ 3371 IC50 = 2230 nM T60529 D0DJ1B 156391 IC50 = 350 nM T60529 D0G7FJ 54677470 IC50 = 1400 nM T60529 D0GY5Z 2244 IC50 = 11400 nM T60529 D0I0EG 44093 Ki = 17000 nM T60529 D0IT2X 2581 IC50 = 13200 nM T60529 D0L6DA 119607 IC50 = 140000 nM T60529 D0M9DC 4614 IC50 = 740 nM T60529 D0N1WU 3308 IC50 = 10300 nM T60529 D0NF1U 64929 IC50 = 950000 nM T60529 D0R1QE 3672 IC50 = 290 nM T60529 D0R1RS 3715 IC50 = 2 nM T60529 D0TG1H 3033 IC50 = 12 nM T60529 D0U5CE 1548943 IC50 = 3800 nM T60529 D0U5QK 1983 IC50 = 200000 nM T60529 D0W9WF 3825 IC50 = 2 nM T60529 D0Y9ZE 4197 IC50 = 4700 nM T60529 D02DYU 9858913 IC50 = 1020 nM T60529 D05FGR 92337 IC50 = 44000 nM T60529 D0AL8T 6444826 IC50 = 600 nM T60529 D0C5DC 72099 IC50 = 2000 nM T60529 D0L4FS 5280961 IC50 = 80000 nM T60529 D0LI1C 44469321 IC50 > 30000 nM T60529 D0U3EP 445154 IC50 = 830 nM T60529 D0U8OD 213053 IC50 = 3300 nM T60529 D0E2TY 71523527 IC50 > 100000 nM T60529 D0F0PK 4711697 IC50 = 4000 nM T60529 D0GY2Z 11394647 IC50 = 48800 nM T60529 D0M6LX 56851703 IC50 > 100000 nM T60529 D0O4QB 3314 IC50 = 11000 nM T60529 D00RSK 9832687 IC50 > 84200 nM T60529 D02OHR 443373 IC50 = 30000 nM T60529 D03NZV 9865808 IC50 = 17800 nM T60529 D05EYG 9799453 IC50 = 1600 nM T60529 D05MCS 44473151 IC50 = 58000 nM T60529 D05REH 71246 IC50 > 50000 nM T60529 D07HBI 132306 IC50 > 100000 nM T60529 D07TZM 115239 IC50 > 20000 nM T60529 D08GRY 3177 IC50 = 59 nM T60529 D09BKE 4553 IC50 = 3000 nM T60529 D0C0JT 4495 IC50 = 3760 nM T60529 D0F8DL 176155 IC50 = 2000 nM T60529 D0N1SU 133021 IC50 = 160 nM T60529 D0O9JX 9851770 IC50 = 140 nM T60529 D0P3KA 60542 IC50 = 250 nM T60529 D0Z5LZ 159271 IC50 > 100000 nM T60529 C8IB3S 3965 IC50 = 6500 nM T60529 CU1X7Z 4237 IC50 = 1.4 nM T60529 C8KED5 4713 IC50 = 1000 nM T60529 CFO1W4 7136 IC50 = 3000 nM T60529 C9KD6A 10189 IC50 = 17800 nM T60529 CV24FH 10228 IC50 > 200000 nM T60529 CCF85O 10774 IC50 > 10000 nM T60529 C4EJ7D 27022 IC50 > 10000 nM T60529 CRVG43 27023 IC50 > 10000 nM T60529 CTY1P6 28566 IC50 > 10000 nM T60529 CMZ01B 37486 IC50 > 10000 nM T60529 CVS6A8 40634 IC50 = 130 nM T60529 CX4FN2 65084 IC50 = 95000 nM T60529 C2FLZ8 65751 IC50 > 30000 nM T60529 CPW9B5 65752 IC50 = 8700 nM T60529 CXE76N 73481 IC50 = 129000 nM T60529 C7L1RO 75522 IC50 > 100000 nM T60529 CHJK85 85393 IC50 > 10000 nM T60529 CZ8U6A 87020 IC50 > 100000 nM T60529 CBED38 100526 IC50 = 18900 nM T60529 C2IRA6 127923 IC50 = 13000 nM T60529 C5GFP0 155948 IC50 > 200000 nM T60529 C70MFQ 159278 IC50 = 72000 nM T60529 CPS7E0 159665 IC50 = 15600 nM T60529 CDC52U 169187 IC50 > 50000 nM T60529 C2KD9Z 171596 IC50 > 50000 nM T60529 C38CSH 176920 IC50 = 3300 nM T60529 C6L5AP 181271 IC50 > 40900 nM T60529 CYWS98 185848 IC50 = 500 nM T60529 CGUW53 196841 IC50 = 28 nM T60529 C2W3TD 263547 IC50 > 10000 nM T60529 C6AKQ8 308411 IC50 = 195740 nM T60529 CM2B0E 377558 IC50 = 1000 nM T60529 C8HA5W 404196 IC50 = 59960 nM T60529 CQCK56 404197 IC50 > 100000 nM T60529 C8BCZ1 404198 IC50 = 23280 nM T60529 CC20HA 404319 IC50 = 167090 nM T60529 C1MKV8 404320 IC50 = 109690 nM T60529 CI1GD8 404323 IC50 = 110270 nM T60529 COU8H0 404325 IC50 = 182190 nM T60529 C56XBC 404376 IC50 = 183500 nM T60529 CFJX25 405488 IC50 = 61730 nM T60529 CD95EA 405490 IC50 = 66410 nM T60529 CJTR17 405491 IC50 = 85130 nM T60529 C01ANL 405559 IC50 = 23150 nM T60529 C3PZ1R 405561 IC50 = 78200 nM T60529 CB60GF 442700 IC50 > 46700 nM T60529 CEI08Y 443378 IC50 = 19000 nM T60529 C65MQP 443639 IC50 = 6400 nM T60529 C2UE5Q 463829 IC50 = 524807.46 nM T60529 CB56XC 480869 IC50 > 100000 nM T60529 C7I8NK 484757 IC50 = 50000 nM T60529 CPJ59X 572426 IC50 = 72000 nM T60529 CCI7B9 572427 IC50 = 88000 nM T60529 CVO51F 591238 IC50 > 30000 nM T60529 CZ7O3I 636928 IC50 = 610 nM T60529 C5YS3J 637775 IC50 = 39200 nM T60529 CQAV61 642530 IC50 = 64300 nM T60529 CMJ91Y 667550 IC50 = 1.9 nM T60529 C28PTM 724576 IC50 = 47910 nM T60529 CW14ZC 827480 IC50 = 17280 nM T60529 C1V7BH 871573 IC50 = 92.2 nM T60529 CMYK57 1500232 IC50 > 50000 nM T60529 C84MXV 1500233 IC50 > 50000 nM T60529 CWNY21 1500235 IC50 > 50000 nM T60529 CI26ZE 1514885 IC50 > 20000 nM T60529 CADY74 1517275 IC50 = 10000 nM T60529 CD89GA 2083607 IC50 = 1000 nM T60529 C1K2QE 2317371 IC50 > 100000 nM T60529 CN9AS5 2756535 IC50 > 100000 nM T60529 CT6W1B 2765724 IC50 > 100000 nM T60529 C9LOJ7 2826057 IC50 = 53700 nM T60529 CQM64G 3037018 IC50 > 20000 nM T60529 CX6D4S 3058754 IC50 = 36000 nM T60529 CXA70K 3080594 IC50 = 234000 nM T60529 CG0MN3 3080635 IC50 > 200000 nM T60529 CP4IL0 3629561 IC50 = 33320 nM T60529 CY2XM7 4226790 IC50 > 10000 nM T60529 C5LQ3D 4322149 IC50 > 20000 nM T60529 CA9X7C 4679898 IC50 = 180 nM T60529 CAKX74 4763851 IC50 = 30760 nM T60529 CJ74EB 4990103 IC50 = 43800 nM T60529 CNPV35 5018304 IC50 = 3 nM T60529 CVT05I 5080393 IC50 > 100000 nM T60529 C0IS9Y 5100138 IC50 > 10000 nM T60529 CDU89L 5195985 IC50 = 82.1 nM T60529 CU4E5S 5273569 IC50 = 524000 nM T60529 CGO6J3 5280372 IC50 = 75000 nM T60529 C1BPI8 5280569 IC50 = 140000 nM T60529 CKC96D 5281232 IC50 = 28000 nM T60529 C0D3PO 5281671 IC50 = 100000 nM T60529 C3VS8X 5316860 IC50 = 36000 nM T60529 CPRI38 5320318 IC50 = 64000 nM T60529 CC3QF0 5321018 IC50 > 200000 nM T60529 CJ8P4T 5352624 IC50 = 115 nM T60529 CH6DT9 5481958 IC50 = 62000 nM T60529 CWS5X0 5481970 IC50 = 14000 nM T60529 C7B1CG 5487413 IC50 = 10000 nM T60529 CS03BA 6255462 IC50 = 25800 nM T60529 C9J6LF 6426663 IC50 = 55100 nM T60529 CF8E2M 6444394 IC50 = 9300 nM T60529 CC97TP 7972918 IC50 = 990 nM T60529 C3BU5H 8566717 IC50 > 100000 nM T60529 CLF8W5 9559931 IC50 = 405960 nM T60529 CB7LR9 9644405 IC50 = 150450 nM T60529 C0NTV6 9795652 IC50 = 29200 nM T60529 CC38MG 9796843 IC50 = 34000 nM T60529 CR7OZ3 9797003 IC50 = 28100 nM T60529 C9MX1U 9797752 IC50 = 27900 nM T60529 C08TVM 9797804 IC50 = 30 nM T60529 C7JYX6 9798239 IC50 = 34300 nM T60529 C24SGI 9798392 IC50 = 11000 nM T60529 CSQD86 9799387 IC50 > 1000000 nM T60529 C1N8HK 9800211 IC50 = 5700 nM T60529 C2XRG4 9800221 IC50 > 1100 nM T60529 CSA4F1 9800270 IC50 = 80 nM T60529 C64NBT 9801204 IC50 = 6200 nM T60529 CV5S6A 9801701 IC50 < 140 nM T60529 CEH9Y2 9808627 IC50 = 138000 nM T60529 CZT7M2 9816662 IC50 > 10000 nM T60529 CC6A2L 9817667 IC50 = 540 nM T60529 CV5Y2H 9818233 IC50 = 3100 nM T60529 C2AKX0 9818254 IC50 = 300000 nM T60529 CQK3E5 9818359 IC50 = 24378.11 nM T60529 C03FBZ 9818888 IC50 = 1120000 nM T60529 CZ0K8H 9819804 IC50 = 36000 nM T60529 C9M2PZ 9820390 IC50 = 265700 nM T60529 C9RST2 9821264 IC50 = 9200 nM T60529 CW37TE 9821646 IC50 > 1000000 nM T60529 CUO02B 9822332 IC50 = 360000 nM T60529 CC75ZO 9822357 IC50 > 91629 nM T60529 C3ZTC7 9822818 IC50 = 3290 nM T60529 CS96DK 9822874 IC50 = 1200 nM T60529 CB0Y6K 9823368 IC50 > 100000 nM T60529 CV7T4Q 9823594 IC50 > 100000 nM T60529 C1E2DV 9826083 IC50 > 80000 nM T60529 CP94CU 9831791 IC50 = 690 nM T60529 CEGR47 9835721 IC50 = 470 nM T60529 CUT4N2 9836619 IC50 = 4200 nM T60529 CISH24 9836698 IC50 = 37000 nM T60529 CZV0R6 9839351 IC50 = 147500 nM T60529 C2TPB6 9839884 IC50 = 18000 nM T60529 CD9YC2 9840237 IC50 > 100000 nM T60529 CTYZ07 9840502 IC50 = 21100 nM T60529 CK65IB 9840638 IC50 > 100000 nM T60529 CBSM70 9840662 IC50 = 84600 nM T60529 C23HSC 9841079 IC50 = 18300 nM T60529 C2NDG3 9841276 IC50 = 33700 nM T60529 CA1YN6 9841715 IC50 > 100000 nM T60529 CA9IV0 9842523 IC50 = 17410 nM T60529 C8Y4ND 9842547 IC50 > 100000 nM T60529 C6U5CF 9842936 IC50 > 1000000 nM T60529 C6HDX1 9842937 IC50 > 1000000 nM T60529 CF15GO 9843089 IC50 = 25500 nM T60529 CJIN69 9843189 IC50 > 10000 nM T60529 C4RSA3 9843356 IC50 = 2800 nM T60529 CMX5B4 9844547 IC50 > 100000 nM T60529 C34IOV 9846219 IC50 = 43700 nM T60529 C94NVU 9846581 IC50 = 1000 nM T60529 CXQ6E3 9858164 IC50 = 140 nM T60529 C49AFB 9861219 IC50 = 116400 nM T60529 CP75VI 9861581 IC50 = 145000 nM T60529 CS6Y5U 9861661 IC50 = 7000 nM T60529 CJLR90 9861712 IC50 > 10000 nM T60529 C5AP3Q 9861854 IC50 > 100000 nM T60529 CV57DI 9861888 IC50 = 47500 nM T60529 CX87MB 9863426 IC50 > 100000 nM T60529 C5NG2Y 9863475 IC50 = 43000 nM T60529 C49BAD 9864100 IC50 > 10000 nM T60529 C2TP7H 9865298 IC50 = 22300 nM T60529 CP4QG9 9865547 IC50 = 2580 nM T60529 C27YKN 9865599 IC50 = 20000 nM T60529 C7ZEH1 9868819 IC50 = 1500 nM T60529 CA43PC 9871042 IC50 > 66000 nM T60529 CSE53Z 9878306 IC50 = 2200 nM T60529 CY1AR6 9880758 IC50 = 31000 nM T60529 CWP06Z 9882419 IC50 = 791100 nM T60529 CP2NZ0 9883585 IC50 = 1 nM T60529 C43HGV 9883653 IC50 = 1000 nM T60529 C1FOR4 9883749 IC50 > 10000 nM T60529 CS6HN1 9883822 IC50 = 2000 nM T60529 C8U7TB 9883880 IC50 = 17000 nM T60529 CYU2N6 9884096 IC50 = 13200 nM T60529 CZF0A2 9884371 IC50 > 100000 nM T60529 CMV92I 9885354 IC50 = 12500 nM T60529 CV0SP3 9901158 IC50 = 36300 nM T60529 CILP75 9901319 IC50 = 4390 nM T60529 CU21FI 9902732 IC50 = 81000 nM T60529 C9ON6P 9902810 IC50 > 100000 nM T60529 C7JE5S 9904089 IC50 > 10000 nM T60529 C2SRN6 9905412 IC50 > 100000 nM T60529 COA31Z 9905676 IC50 = 5100 nM T60529 C2YDI0 9905875 IC50 > 8600 nM T60529 CAH7V1 9906472 IC50 = 5100 nM T60529 C4YE6S 9906813 IC50 = 52600 nM T60529 C4P5DV 9907758 IC50 = 2200 nM T60529 CG8P5T 9908624 IC50 = 1000 nM T60529 C2T6IY 9908677 IC50 = 29000 nM T60529 C1SEB7 9909016 IC50 > 100000 nM T60529 CQ83VI 9909642 IC50 < 140 nM T60529 CD0J1F 9918457 IC50 = 500 nM T60529 C0Y5BR 9922118 IC50 = 1080 nM T60529 CE2LZ0 9922659 IC50 = 25600 nM T60529 CWJH86 9922739 IC50 = 4.9 nM T60529 CZ0IQ2 9923656 IC50 > 50000 nM T60529 CSU35P 9924251 IC50 > 100000 nM T60529 C06GJS 9925288 IC50 > 58000 nM T60529 C5C9DS 9925578 IC50 > 10000 nM T60529 C42GTD 9926659 IC50 = 20000 nM T60529 CR8TW5 9927594 IC50 > 100000 nM T60529 C2QSC1 9927613 IC50 = 1300 nM T60529 CK71LW 9927909 IC50 > 100000 nM T60529 CG1C3L 9927912 IC50 = 1320 nM T60529 CY1F3R 9928047 IC50 = 330 nM T60529 CXY6V4 9928340 IC50 = 13600 nM T60529 C2OUH1 9928381 IC50 = 6998.42 nM T60529 C70GRD 9928539 IC50 > 50000 nM T60529 COE0X2 9928728 IC50 > 100000 nM T60529 C2CJ4G 9929140 IC50 > 10000000 nM T60529 C8Z3SJ 9929308 IC50 = 6300 nM T60529 CS7EB8 9929562 IC50 < 700 nM T60529 CT0HB7 9929697 IC50 = 830 nM T60529 C8N4FQ 9930747 IC50 > 10000 nM T60529 CHS01T 9930803 IC50 = 11600 nM T60529 C9HQ1Z 9931215 IC50 = 39300 nM T60529 CUVI39 9932045 IC50 = 590 nM T60529 CS2ZH4 9932828 IC50 = 5600 nM T60529 C6QPN2 9933112 IC50 > 100000 nM T60529 CJ4AV0 9933456 IC50 > 100000 nM T60529 C97YOJ 9936231 IC50 > 66000 nM T60529 CA7M2V 9942292 IC50 = 22200 nM T60529 C6RQW1 9945282 IC50 = 10 nM T60529 CU6J7M 9945403 IC50 > 100000 nM T60529 CXK27R 9946200 IC50 > 100000 nM T60529 CF9QL0 9946917 IC50 > 10000 nM T60529 CH7ZK2 9947111 IC50 > 100000 nM T60529 CWU4Y1 9947165 IC50 > 100000 nM T60529 CQC75N 9947305 IC50 = 723000 nM T60529 CYQF10 9947309 IC50 > 100000 nM T60529 CIC92Y 9947371 IC50 > 1000000 nM T60529 CKWB53 9947925 IC50 = 550 nM T60529 C4WC8T 9948569 IC50 = 10000 nM T60529 CEH6M2 9948850 IC50 = 18400 nM T60529 CYOR40 9948878 IC50 = 45600 nM T60529 C42BFH 9949984 IC50 = 42364.3 nM T60529 C0GC2F 9950666 IC50 > 100000 nM T60529 C87QWC 9950669 IC50 = 3000 nM T60529 CUV05Z 9954100 IC50 > 100000 nM T60529 CL1W0Y 9954883 IC50 = 8490 nM T60529 CAU01B 9957131 IC50 > 100000 nM T60529 C04ZJC 9965352 IC50 = 100000 nM T60529 CZN2B4 9966560 IC50 = 94500 nM T60529 CMF25N 9967049 IC50 = 59000 nM T60529 C25VMC 9967345 IC50 = 42000 nM T60529 CQX38P 9967467 IC50 = 118000 nM T60529 CS8VF5 9967867 IC50 > 100000 nM T60529 CA8E7F 9968075 IC50 > 125000 nM T60529 CP5O2E 9969153 IC50 = 60000 nM T60529 C5XM8F 9969968 IC50 > 100000 nM T60529 C4K0IL 9970134 IC50 = 338000 nM T60529 C4AUM2 9973893 IC50 > 100000 nM T60529 CDA38U 9987332 IC50 = 59000 nM T60529 CO68GP 9993267 IC50 = 51 nM T60529 CQO56T 9993978 IC50 > 100000 nM T60529 CJ9E2P 9998267 IC50 > 30000 nM T60529 CWY7U3 10001441 IC50 = 5860 nM T60529 C6FM2Z 10001804 IC50 = 5740 nM T60529 C26QHZ 10005638 IC50 > 80000 nM T60529 CMJH05 10016051 IC50 = 500000 nM T60529 CTR6H1 10019555 IC50 = 34000 nM T60529 CLEY67 10019929 IC50 > 20000 nM T60529 CC7M1T 10020588 IC50 > 100000 nM T60529 CY4K1P 10021211 IC50 = 55 nM T60529 C05TFO 10021647 IC50 = 17300 nM T60529 CG49LP 10021928 IC50 > 100000 nM T60529 CQH70M 10022177 IC50 > 100000 nM T60529 C0UN1I 10022305 IC50 = 250 nM T60529 CC03QH 10024599 IC50 = 400 nM T60529 C7IEL6 10037656 IC50 = 280 nM T60529 CDE7V9 10038859 IC50 = 100000 nM T60529 C4CD3P 10040599 IC50 = 17000 nM T60529 C1EAZ3 10041271 IC50 > 100000 nM T60529 CI6F3U 10044786 IC50 > 100000 nM T60529 CIS0T3 10046006 IC50 = 1420 nM T60529 C9C4IM 10046378 IC50 = 5500 nM T60529 CT54KN 10047220 IC50 > 250000 nM T60529 CRK0M8 10051539 IC50 = 384000 nM T60529 C8WTM1 10064144 IC50 = 1510 nM T60529 CS40HT 10064410 IC50 = 1200 nM T60529 C58CDE 10068193 IC50 > 10000 nM T60529 C7U9DB 10069246 IC50 = 81800 nM T60529 C0OQF8 10071029 IC50 = 3600 nM T60529 CJN53X 10084869 IC50 = 159720 nM T60529 CI9MW1 10087345 IC50 = 12000 nM T60529 CSA7R2 10088207 IC50 = 47500 nM T60529 CCQ28U 10088506 IC50 > 100000 nM T60529 CW05LQ 10090654 IC50 > 100000 nM T60529 C9HR8U 10095369 IC50 > 100000 nM T60529 C7IEF9 10095474 IC50 = 4300 nM T60529 CHV67O 10108931 IC50 > 90000 nM T60529 C92OBR 10109075 IC50 > 100000 nM T60529 CW3J9B 10109361 IC50 > 60000 nM T60529 C90KPZ 10109982 IC50 > 10000 nM T60529 CF2L8T 10110298 IC50 = 78000 nM T60529 C67SQN 10110427 IC50 = 1320 nM T60529 CRKC39 10110822 IC50 = 21200 nM T60529 CO98VP 10113620 IC50 > 10000 nM T60529 CIF46A 10118686 IC50 > 100000 nM T60529 C0QF5M 10131479 IC50 = 5000 nM T60529 CBDU01 10133653 IC50 > 10000 nM T60529 CU2TS5 10133741 IC50 = 22800 nM T60529 CPEL28 10133748 IC50 > 100000 nM T60529 C64UXL 10134425 IC50 = 4600 nM T60529 CO0EY4 10134426 IC50 = 3200 nM T60529 CL4ZX6 10135355 IC50 = 13800 nM T60529 CUC48F 10136509 IC50 = 49000 nM T60529 C62HSP 10138952 IC50 = 22803.42 nM T60529 C39FVT 10154719 IC50 > 100000 nM T60529 C3ALT5 10155221 IC50 > 100000 nM T60529 CU0QS9 10155469 IC50 = 1600 nM T60529 CCFX37 10155819 IC50 = 19300 nM T60529 CXL35F 10156006 IC50 > 50000 nM T60529 C89SFQ 10156048 IC50 > 100000 nM T60529 CGY3U6 10156369 IC50 = 1000 nM T60529 C75HBA 10156402 IC50 > 10000 nM T60529 CYXL62 10156660 IC50 = 33900 nM T60529 CY8WB7 10156700 IC50 > 1000 nM T60529 C97MLG 10156720 IC50 = 84000 nM T60529 CT16EK 10157135 IC50 > 100000 nM T60529 C0LZU6 10157427 IC50 = 3000 nM T60529 C8EP6N 10157624 IC50 > 10000 nM T60529 C91PJR 10157862 IC50 > 100000 nM T60529 CB8PS0 10158806 IC50 = 570 nM T60529 CN62VZ 10159879 IC50 = 5800 nM T60529 CG6FC7 10172237 IC50 > 10000 nM T60529 C3EFY5 10177578 IC50 = 6010 nM T60529 CE9PV5 10177830 IC50 > 10000 nM T60529 CP3C8N 10177845 IC50 > 1000000 nM T60529 C1O8JD 10178729 IC50 = 380 nM T60529 C4U5VF 10179720 IC50 = 18900 nM T60529 CPTS56 10179876 IC50 = 15500 nM T60529 C50MBD 10180742 IC50 > 100000 nM T60529 C73DEB 10181405 IC50 > 100000 nM T60529 CK05GP 10183636 IC50 = 35196.54 nM T60529 CG2Y1Q 10199429 IC50 = 58000 nM T60529 C9VW0L 10199643 IC50 = 31000 nM T60529 C5WB6K 10199764 IC50 = 25900 nM T60529 CN5O6D 10199832 IC50 = 18100 nM T60529 C7V6HN 10200639 IC50 = 1000 nM T60529 COEJ03 10200640 IC50 < 300 nM T60529 CT4I3O 10200696 IC50 > 10000 nM T60529 CZL86N 10200745 IC50 = 76000 nM T60529 C10MGH 10200861 IC50 > 100000 nM T60529 CXA45O 10200928 IC50 = 82000 nM T60529 CBD58L 10201258 IC50 = 36559.48 nM T60529 C5GSU9 10201259 IC50 = 16595.87 nM T60529 CLI4G2 10201726 IC50 > 100000 nM T60529 C0CDF4 10201744 IC50 = 3000 nM T60529 CIG42D 10202758 IC50 > 100000 nM T60529 CS4Y1F 10221647 IC50 > 100000 nM T60529 C0E4ZO 10221859 IC50 = 6902.4 nM T60529 C12ZGN 10222021 IC50 > 10000 nM T60529 CW17QB 10222707 IC50 = 31300 nM T60529 C1OH3T 10222861 IC50 > 10000 nM T60529 C6JLS5 10223461 IC50 = 1360 nM T60529 CEKL34 10224978 IC50 = 17400 nM T60529 CK31YH 10224979 IC50 = 31200 nM T60529 CCT79E 10227082 IC50 > 100000 nM T60529 C1KF3U 10237369 IC50 = 40 nM T60529 CU8G6W 10244247 IC50 = 3300 nM T60529 CRF02L 10246625 IC50 > 45000 nM T60529 C9Q3GN 10251114 IC50 = 3000 nM T60529 C1YF7W 10255326 IC50 > 500000 nM T60529 C1R9VI 10265882 IC50 = 42 nM T60529 COQ0I9 10267703 IC50 = 740 nM T60529 CRVU30 10268555 IC50 = 1300 nM T60529 C5U6ZL 10269056 IC50 = 63000 nM T60529 COG84H 10269175 IC50 = 8100 nM T60529 CDJO97 10269858 IC50 = 800 nM T60529 C4D1AW 10270798 IC50 > 10000 nM T60529 CRP52C 10271231 IC50 > 1000000 nM T60529 CKZ72U 10271396 IC50 = 29500 nM T60529 CNJ96H 10272113 IC50 > 100000 nM T60529 CU45JL 10272435 IC50 = 40000 nM T60529 CQ6ZK8 10273159 IC50 = 1190 nM T60529 C15AKU 10273161 IC50 > 100000 nM T60529 CVQ9R1 10273329 IC50 > 100000 nM T60529 CCT59Q 10273651 IC50 > 100000 nM T60529 CJE46B 10292387 IC50 > 100000 nM T60529 CV2OS0 10292572 IC50 > 100000 nM T60529 C3GB8J 10292693 IC50 = 13000 nM T60529 C19RZV 10293184 IC50 > 1000000 nM T60529 CG1I7N 10293242 IC50 = 89000 nM T60529 CX3J6F 10294269 IC50 = 1200 nM T60529 CA37EH 10294458 IC50 = 1070 nM T60529 CYW2V3 10294501 IC50 > 100000 nM T60529 C9JN8Q 10294921 IC50 > 100000 nM T60529 CR02XQ 10295072 IC50 > 10000 nM T60529 C3FL9K 10295633 IC50 > 80000 nM T60529 C2QA8P 10296709 IC50 = 65 nM T60529 C3X7IN 10316629 IC50 = 5700 nM T60529 CK1WP4 10316962 IC50 > 50000 nM T60529 C1OSM9 10318787 IC50 = 1860 nM T60529 CITV57 10319221 IC50 = 10800 nM T60529 C1C4NS 10330671 IC50 = 13000 nM T60529 C0K1GF 10335077 IC50 = 25900 nM T60529 C1LZ7Y 10335263 IC50 = 1000 nM T60529 CWG32C 10336743 IC50 = 28973.44 nM T60529 CB06KL 10336873 IC50 > 100000 nM T60529 C7AY2L 10337564 IC50 = 3000 nM T60529 CCV82I 10339513 IC50 = 5800 nM T60529 CA3XB0 10339727 IC50 = 58000 nM T60529 C1REP8 10355223 IC50 = 500 nM T60529 CLID50 10359269 IC50 = 6500 nM T60529 CM01BR 10359484 IC50 = 96100 nM T60529 C6P9HD 10360345 IC50 = 880 nM T60529 CJG7W4 10360688 IC50 = 18 nM T60529 CU5Y3X 10361821 IC50 = 32700 nM T60529 CI42KJ 10363144 IC50 = 300 nM T60529 CX8ZA1 10363491 IC50 > 10000 nM T60529 CKH1A6 10381453 IC50 > 100000 nM T60529 C9CJY4 10381501 IC50 = 1000 nM T60529 CH8WQ5 10381921 IC50 = 258110 nM T60529 CDB2Z0 10383075 IC50 = 2700 nM T60529 C7VP2Q 10385170 IC50 = 8200 nM T60529 CI67YJ 10385715 IC50 > 50000 nM T60529 C9SPO1 10385880 IC50 = 22500 nM T60529 CY4W2C 10386019 IC50 > 10000 nM T60529 CA8B5T 10390073 IC50 > 80000 nM T60529 CSR51N 10403254 IC50 > 100000 nM T60529 CA7QF5 10405126 IC50 > 100000 nM T60529 CFL72P 10405693 IC50 > 100000 nM T60529 C5JHI0 10406427 IC50 = 14400 nM T60529 CFXL12 10406946 IC50 > 100000 nM T60529 CP40MA 10407440 IC50 = 5800 nM T60529 C17TBC 10407720 IC50 = 22300 nM T60529 C9SRX6 10408088 IC50 > 100000 nM T60529 C39ISW 10408494 IC50 = 1130 nM T60529 C52MXI 10413126 IC50 = 14000 nM T60529 CG8T1K 10414246 IC50 = 3700 nM T60529 C2L8RQ 10424013 IC50 = 350 nM T60529 CA3X7E 10424186 IC50 = 970 nM T60529 CA1S7I 10425292 IC50 = 2280 nM T60529 CGU4Q8 10425834 IC50 > 100000 nM T60529 CW6H4S 10426661 IC50 > 100000 nM T60529 CP57LS 10426884 IC50 > 100000 nM T60529 CQ7Z6C 10428486 IC50 = 4400 nM T60529 C3NK6J 10430343 IC50 > 1000000 nM T60529 CA24ER 10433546 IC50 > 100000 nM T60529 C1T4PM 10446327 IC50 = 210 nM T60529 C65BPM 10447425 IC50 > 100000 nM T60529 C72ERI 10448879 IC50 > 100000 nM T60529 CIMC74 10449604 IC50 = 98000 nM T60529 CVF6I8 10452350 IC50 = 577000 nM T60529 CLV8C6 10452657 IC50 > 100000 nM T60529 CQ94JT 10453591 IC50 = 69000 nM T60529 CGD93Y 10457034 IC50 > 66000 nM T60529 C1WM2V 10459826 IC50 > 10 nM T60529 CB50TO 10471014 IC50 = 10500 nM T60529 C3TK7X 10472597 IC50 > 100000 nM T60529 C7DT1E 10476542 IC50 = 3752 nM T60529 COL4Z0 10476930 IC50 = 3800 nM T60529 CLP06F 10493616 IC50 = 2000 nM T60529 C3ZM1X 10494600 IC50 > 10000 nM T60529 CMS87O 10497881 IC50 = 580 nM T60529 C4CRG9 10498736 IC50 = 740 nM T60529 C5CZB7 10498979 IC50 = 5100 nM T60529 CHQ85J 10499452 IC50 > 100000 nM T60529 CZD6A8 10500038 IC50 > 1000000 nM T60529 CW9EQ6 10500466 IC50 > 100000 nM T60529 CC0Z4F 10500696 IC50 > 100000 nM T60529 CPO37N 10500778 IC50 = 500 nM T60529 CZ7IX5 10500888 IC50 = 53500 nM T60529 C65HEP 10501037 IC50 > 100000 nM T60529 CMJ08V 10501190 IC50 = 23000 nM T60529 CU8KR5 10501652 IC50 = 5000 nM T60529 C6O1UH 10501957 IC50 = 12000 nM T60529 C2QN6Y 10501958 IC50 > 1000000 nM T60529 CE4S1Y 10502827 IC50 = 8600 nM T60529 CR4OK6 10504537 IC50 > 100000 nM T60529 CI16BX 10506935 IC50 > 100000 nM T60529 CI6F7S 10516483 IC50 = 95 nM T60529 CCO02A 10517413 IC50 = 290 nM T60529 C8JTN1 10518222 IC50 = 1450 nM T60529 CGC62Z 10519259 IC50 > 100000 nM T60529 CF57BP 10520447 IC50 > 100000 nM T60529 CO6D8P 10520508 IC50 > 100000 nM T60529 C9WDP7 10520866 IC50 = 710 nM T60529 CZ4MX2 10521318 IC50 = 60 nM T60529 CL2WV6 10521660 IC50 = 1700 nM T60529 CLK73W 10521710 IC50 = 20000 nM T60529 CLZ4D8 10522463 IC50 > 100000 nM T60529 CGMA31 10522592 IC50 = 920 nM T60529 CS3L6E 10522977 IC50 = 4000 nM T60529 CQ3S6J 10523033 IC50 = 3800 nM T60529 C35MKT 10523190 IC50 > 100000 nM T60529 CCM67S 10523255 IC50 > 100000 nM T60529 CB2EZ0 10523413 IC50 = 8200 nM T60529 CXO9S1 10524261 IC50 > 100000 nM T60529 C52QXF 10524370 IC50 = 1700 nM T60529 CU7Z4M 10524532 IC50 = 18000 nM T60529 C17KQI 10524587 IC50 > 100000 nM T60529 C0N4YM 10524857 IC50 > 100000 nM T60529 CA4TO8 10524898 IC50 > 100000 nM T60529 CEO49Q 10524951 IC50 > 100000 nM T60529 CS14IM 10525575 IC50 > 10000 nM T60529 CTKM86 10525659 IC50 = 8800 nM T60529 CRI9N3 10526696 IC50 > 100000 nM T60529 CF1PX9 10526904 IC50 > 100000 nM T60529 C54DWE 10541466 IC50 = 2500 nM T60529 C8YI0Q 10541610 IC50 > 100000 nM T60529 C58BNM 10543451 IC50 > 100000 nM T60529 CN6M2J 10543472 IC50 = 15000 nM T60529 CNQ03M 10544389 IC50 = 10889.3 nM T60529 C4AV8Q 10545354 IC50 = 3981.07 nM T60529 C47RFN 10545379 IC50 = 10399.2 nM T60529 CIB05E 10545620 IC50 > 50000 nM T60529 C4N8QO 10545724 IC50 > 100000 nM T60529 C9UB1K 10546170 IC50 > 100000 nM T60529 CQ32BJ 10546382 IC50 > 100000 nM T60529 C0JP5I 10546567 IC50 > 100000 nM T60529 C1TPD4 10547228 IC50 > 100000 nM T60529 C2YV6X 10547351 IC50 = 14600 nM T60529 C8U3CE 10548520 IC50 > 100000 nM T60529 CICG32 10549411 IC50 = 800 nM T60529 C1H7JD 10549466 IC50 = 1210 nM T60529 CBH0K1 10549551 IC50 > 100000 nM T60529 C62ITD 10549657 IC50 > 100000 nM T60529 C1YLO7 10549795 IC50 = 2500 nM T60529 CIR1X4 10563380 IC50 = 3500 nM T60529 CCNY05 10564674 IC50 = 16000 nM T60529 C6M5YN 10567176 IC50 > 10000 nM T60529 C9SOC2 10568310 IC50 = 20000 nM T60529 CP6JX9 10568417 IC50 > 100000 nM T60529 CM89NX 10569712 IC50 = 5 nM T60529 CU1RH9 10569839 IC50 > 100000 nM T60529 CG8HY7 10569949 IC50 > 50000 nM T60529 CS74PE 10570051 IC50 > 100000 nM T60529 CU5GB2 10570135 IC50 = 570 nM T60529 CN2W5O 10570444 IC50 > 100000 nM T60529 CZ38CW 10570970 IC50 > 100000 nM T60529 C6FAO5 10571335 IC50 > 100000 nM T60529 CN1TG0 10571627 IC50 = 3700 nM T60529 C9PT5C 10571870 IC50 > 100000 nM T60529 CGVM06 10572070 IC50 = 36000 nM T60529 CLBY56 10572128 IC50 = 1900 nM T60529 CADV12 10572129 IC50 = 67700 nM T60529 CQAJ45 10572620 IC50 > 100000 nM T60529 C5WPQ6 10573666 IC50 = 15400 nM T60529 CYJ9V0 10574324 IC50 = 16400 nM T60529 CX17PF 10574332 IC50 > 100000 nM T60529 C5HXO6 10574480 IC50 = 17100 nM T60529 CUY9N4 10574542 IC50 > 100000 nM T60529 C1ECI8 10574823 IC50 = 400 nM T60529 C6LSX4 10575260 IC50 = 1560 nM T60529 CDA0F5 10575436 IC50 = 77000 nM T60529 CHM8O7 10576610 IC50 > 100000 nM T60529 C2P3EL 10576988 IC50 > 100000 nM T60529 C3P8XQ 10590357 IC50 = 340 nM T60529 C2UPC7 10592313 IC50 = 4100 nM T60529 C3ZQ9G 10592466 IC50 = 200 nM T60529 C0PNH9 10592721 IC50 = 650 nM T60529 CQ5HY9 10594681 IC50 > 100000 nM T60529 CI6WX3 10594776 IC50 > 100000 nM T60529 CEH6S3 10594921 IC50 = 2700 nM T60529 CV61CE 10594959 IC50 = 5000 nM T60529 C32XIL 10595453 IC50 > 100000 nM T60529 CF8JP2 10596233 IC50 = 14500 nM T60529 C48WTA 10596725 IC50 > 100000 nM T60529 C9S6WU 10596883 IC50 > 100000 nM T60529 CTO61I 10597216 IC50 > 100000 nM T60529 CR9D4F 10597571 IC50 > 100000 nM T60529 C23IOF 10598294 IC50 > 100000 nM T60529 CY29BU 10598409 IC50 = 91000 nM T60529 CN03KT 10598578 IC50 = 6330 nM T60529 C8DT5Q 10598702 IC50 > 100000 nM T60529 CCY5L1 10600544 IC50 > 100000 nM T60529 CW8G7F 10600662 IC50 = 2740 nM T60529 CUZ7B1 10615540 IC50 = 400 nM T60529 CT5S2N 10616370 IC50 = 30000 nM T60529 CG2A5Z 10616776 IC50 = 8100 nM T60529 C37IWY 10617890 IC50 = 10789.47 nM T60529 C8YQ6N 10618038 IC50 > 100000 nM T60529 CWN28D 10618802 IC50 = 300 nM T60529 C8KLQ0 10619035 IC50 = 1400 nM T60529 C5GWB7 10619274 IC50 > 100000 nM T60529 CV5WA8 10619336 IC50 = 55000 nM T60529 C49FXO 10619703 IC50 > 100000 nM T60529 CH4M5Z 10619979 IC50 > 10000 nM T60529 C3U7ME 10620295 IC50 > 1000000 nM T60529 CJ8X1M 10620528 IC50 > 100000 nM T60529 CEF30U 10620563 IC50 > 100000 nM T60529 C8T6QN 10620570 IC50 > 100000 nM T60529 CGN4X1 10620694 IC50 > 100000 nM T60529 C27RKQ 10621114 IC50 > 100000 nM T60529 CX34BP 10621294 IC50 > 100000 nM T60529 CSMA50 10621472 IC50 = 42200 nM T60529 CP63ZJ 10621562 IC50 > 100000 nM T60529 CGV75S 10621593 IC50 = 52000 nM T60529 CRXA24 10621689 IC50 = 27600 nM T60529 C0I4UK 10622186 IC50 = 70700 nM T60529 C7Z3AE 10623138 IC50 > 100000 nM T60529 C6Z3DW 10623232 IC50 > 100000 nM T60529 C8C2XD 10623316 IC50 = 3540 nM T60529 CD51RW 10623882 IC50 > 100000 nM T60529 C9NQP1 10624176 IC50 > 100000 nM T60529 C5N1ZT 10637982 IC50 > 100000 nM T60529 CXJN98 10638180 IC50 = 2500 nM T60529 C5OIE6 10639657 IC50 > 1000 nM T60529 C5QJT8 10641092 IC50 > 100000 nM T60529 C2H9QZ 10641380 IC50 > 100000 nM T60529 C08ESX 10641720 IC50 > 100000 nM T60529 CJIL86 10642557 IC50 = 100 nM T60529 CB63LQ 10642954 IC50 > 100000 nM T60529 CYWU12 10643086 IC50 = 480 nM T60529 CV01MH 10643308 IC50 > 100000 nM T60529 CS9X7O 10643550 IC50 > 10000 nM T60529 CLZ52N 10643725 IC50 > 100000 nM T60529 C6X3QR 10644259 IC50 = 140 nM T60529 CMA47V 10644309 IC50 = 16500 nM T60529 C4KF7S 10644380 IC50 > 100000 nM T60529 C5E1UO 10644539 IC50 = 170 nM T60529 CP9O6S 10644759 IC50 = 1600 nM T60529 C0Z2LW 10645180 IC50 = 1800 nM T60529 C3DJ8A 10645484 IC50 > 100000 nM T60529 C4I8CE 10646043 IC50 = 674000 nM T60529 C0EAM8 10646465 IC50 > 100000 nM T60529 CE98OM 10646723 IC50 = 12900 nM T60529 CGO89K 10660176 IC50 > 100000 nM T60529 C9N8EC 10662676 IC50 > 10000 nM T60529 C2UCE6 10663006 IC50 > 100000 nM T60529 C2X9JN 10663080 IC50 = 5100 nM T60529 CG9VC6 10663833 IC50 > 100000 nM T60529 C6Z5MJ 10664116 IC50 > 100000 nM T60529 C4JQH6 10664141 IC50 = 4500 nM T60529 C65CUY 10664448 IC50 > 100000 nM T60529 CF7I3B 10664738 IC50 > 100000 nM T60529 CRD7N4 10665073 IC50 = 1900 nM T60529 CMZW27 10665242 IC50 = 899.5 nM T60529 CN1I8K 10665362 IC50 > 100000 nM T60529 C08GOU 10665504 IC50 > 100000 nM T60529 CCB67N 10666170 IC50 = 17000 nM T60529 C94OSF 10666215 IC50 > 100000 nM T60529 CYU03I 10666285 IC50 > 100000 nM T60529 CN58GZ 10666572 IC50 = 37068.07 nM T60529 CX92LU 10666704 IC50 = 209000 nM T60529 CP1H7C 10667040 IC50 > 100000 nM T60529 CQUE64 10667216 IC50 = 37700 nM T60529 CTY5Z0 10667341 IC50 = 310 nM T60529 C2B4UE 10667766 IC50 = 1499.68 nM T60529 CBU0Z6 10667777 IC50 = 830 nM T60529 C63ZDJ 10668272 IC50 > 100000 nM T60529 CF39UA 10668540 IC50 = 24100 nM T60529 C5BL8W 10668860 IC50 = 29800 nM T60529 CQ8G9S 10668927 IC50 > 100000 nM T60529 C72XSN 10669268 IC50 > 100000 nM T60529 C8R1WI 10669397 IC50 = 8710 nM T60529 C3AIJ5 10669481 IC50 = 129600 nM T60529 C0L1YR 10669511 IC50 = 7840 nM T60529 CO7MC2 10670044 IC50 > 100000 nM T60529 CC9KU0 10670425 IC50 > 30000 nM T60529 CF4ZD1 10670953 IC50 > 100000 nM T60529 C6CS5M 10671076 IC50 > 1000000 nM T60529 CW0M4E 10685712 IC50 = 70 nM T60529 CKZ6D7 10686987 IC50 > 100000 nM T60529 C5OA4S 10688075 IC50 = 13396.77 nM T60529 C5NZ4I 10688742 IC50 > 100000 nM T60529 CF5XO3 10688810 IC50 > 100000 nM T60529 CRWF25 10689255 IC50 = 6934.26 nM T60529 C7IMK5 10689263 IC50 < 1000 nM T60529 CIMT60 10689279 IC50 > 50000 nM T60529 C2R0UI 10690316 IC50 > 10000 nM T60529 CA9B7R 10690364 IC50 = 93300 nM T60529 CS4QA8 10690636 IC50 > 1000000 nM T60529 C9DUH1 10691290 IC50 = 302000 nM T60529 C58BDY 10691358 IC50 > 100000 nM T60529 CHO5U6 10692230 IC50 = 71600 nM T60529 C6LDV7 10692403 IC50 > 100000 nM T60529 C02IYT 10692761 IC50 = 15200 nM T60529 CX93TR 10693268 IC50 > 1000000 nM T60529 C6YVW5 10693269 IC50 = 82000 nM T60529 CI9CB2 10693380 IC50 > 100000 nM T60529 CPU6N3 10694708 IC50 > 100000 nM T60529 CX65EM 10695000 IC50 = 8980 nM T60529 CF4G6H 10708915 IC50 = 1810 nM T60529 CDPT71 10709447 IC50 = 5000 nM T60529 C1WR8U 10710181 IC50 = 35 nM T60529 CLK87B 10710312 IC50 > 100000 nM T60529 C7HT2G 10710438 IC50 > 100000 nM T60529 CQOD76 10710474 IC50 = 2000 nM T60529 CE6L3I 10711484 IC50 = 6606.93 nM T60529 CT78PA 10711485 IC50 = 49300 nM T60529 CFAO45 10712340 IC50 > 100000 nM T60529 CX5I9C 10712958 IC50 = 15310.87 nM T60529 CJR8V5 10713528 IC50 = 265000 nM T60529 CBM05Q 10714139 IC50 > 50000 nM T60529 C56ECJ 10714428 IC50 > 100000 nM T60529 CU20OI 10714590 IC50 = 1800 nM T60529 CWK7C1 10714907 IC50 > 100000 nM T60529 C54WCH 10715239 IC50 > 1000000 nM T60529 C03QYS 10715523 IC50 > 100000 nM T60529 CEZK47 10715707 IC50 > 10000 nM T60529 CE7M6G 10716372 IC50 = 4690 nM T60529 CSHM17 10716420 IC50 > 100000 nM T60529 CAZ14N 10716484 IC50 > 100000 nM T60529 C89XSQ 10717305 IC50 = 410 nM T60529 C2ICZ5 10717364 IC50 > 100000 nM T60529 CB0A2M 10729933 IC50 = 25000 nM T60529 CE4GJ6 10734248 IC50 = 56500 nM T60529 CZD32K 10735037 IC50 > 100000 nM T60529 CLQ29C 10737761 IC50 = 100 nM T60529 CPQ73G 10738225 IC50 > 100000 nM T60529 C8WKH3 10738721 IC50 > 100000 nM T60529 CB4Y8S 10738786 IC50 > 100000 nM T60529 CM8DE5 10738921 IC50 > 100000 nM T60529 C2O5VB 10739009 IC50 > 100000 nM T60529 C8Q9WG 10739510 IC50 = 3000 nM T60529 C8TQ2M 10740301 IC50 > 100000 nM T60529 C2L9KP 10740567 IC50 > 100000 nM T60529 CFAL86 10740669 IC50 = 32000 nM T60529 CF6QR7 10741315 IC50 = 296000 nM T60529 C4UQ2F 10741367 IC50 > 100000 nM T60529 CNSW35 10741533 IC50 > 100000 nM T60529 CCDT10 10742004 IC50 > 1000000 nM T60529 C14GVA 10742263 IC50 = 2910 nM T60529 C79QXL 10742264 IC50 = 67000 nM T60529 C4JNI5 10746383 IC50 = 5200 nM T60529 CJR19I 10757665 IC50 = 45 nM T60529 C31ZYT 10758665 IC50 = 11000 nM T60529 CKJB53 10758721 IC50 = 11587.77 nM T60529 C41VSC 10759467 IC50 = 4040 nM T60529 CI9LE3 10759852 IC50 = 12200 nM T60529 CEX12Q 10759876 IC50 = 43451.02 nM T60529 CE8TP5 10760536 IC50 > 100000 nM T60529 C34ECZ 10760894 IC50 = 3100 nM T60529 CT9U8B 10760960 IC50 = 140 nM T60529 CW85FZ 10761459 IC50 > 100000 nM T60529 CUB65A 10761664 IC50 > 100000 nM T60529 CYH42G 10762072 IC50 > 100000 nM T60529 CA9Y7S 10762141 IC50 > 100000 nM T60529 CZ12TA 10762494 IC50 > 100000 nM T60529 C3VNE9 10763435 IC50 = 8700 nM T60529 CL91JT 10764155 IC50 > 100000 nM T60529 C43ANY 10764356 IC50 = 930 nM T60529 CWD6R8 10765040 IC50 = 29800 nM T60529 CY62TN 10765111 IC50 = 77700 nM T60529 CQ1YE3 10765731 IC50 > 100000 nM T60529 C2O5CV 10765773 IC50 = 4500 nM T60529 CHK8S2 10766586 IC50 > 100000 nM T60529 CN0CO3 10781432 IC50 = 800 nM T60529 CWM20X 10782440 IC50 = 19000 nM T60529 CG5EO7 10783872 IC50 > 1000 nM T60529 C1SAW6 10783884 IC50 = 27000 nM T60529 CT81VO 10784091 IC50 > 100000 nM T60529 CIFQ86 10784411 IC50 = 5 nM T60529 CNB21H 10784589 IC50 > 100000 nM T60529 CXE17N 10784741 IC50 > 100000 nM T60529 CJ8BO1 10784838 IC50 = 9200 nM T60529 CAE0J1 10786069 IC50 > 100000 nM T60529 C54TIZ 10786081 IC50 > 10000 nM T60529 C4K0GX 10786241 IC50 > 100000 nM T60529 CE5Z1V 10786868 IC50 > 10000 nM T60529 C1IZB3 10786954 IC50 > 100000 nM T60529 CA9U0M 10786970 IC50 > 100000 nM T60529 C37NKS 10786971 IC50 < 1 nM T60529 CLD35X 10787338 IC50 = 17900 nM T60529 CYRC45 10787698 IC50 = 1100 nM T60529 C0X7ME 10787761 IC50 = 28200 nM T60529 CL6I5P 10787918 IC50 > 100000 nM T60529 CZTL42 10789231 IC50 = 5000 nM T60529 C1LRD4 10789363 IC50 > 100000 nM T60529 CA17RT 10799759 IC50 > 100000 nM T60529 CU80LF 10802365 IC50 = 20000 nM T60529 CM13QH 10804032 IC50 > 100000 nM T60529 CO8XJ4 10805003 IC50 > 100000 nM T60529 CSYE98 10807025 IC50 > 50000 nM T60529 CPYI68 10807315 IC50 > 100000 nM T60529 CGP30T 10807353 IC50 = 2300 nM T60529 C32KJP 10807549 IC50 = 2700 nM T60529 C8JM6A 10808251 IC50 = 13182.57 nM T60529 CPA3M7 10808453 IC50 > 100000 nM T60529 CS3L2R 10809519 IC50 > 100000 nM T60529 C1DYX5 10809854 IC50 > 1000000 nM T60529 C4CBE7 10809855 IC50 > 1000000 nM T60529 C4IZ1J 10809969 IC50 > 100000 nM T60529 C1VG3L 10810038 IC50 > 100000 nM T60529 CXEV84 10810080 IC50 > 100000 nM T60529 C69ZEY 10810604 IC50 = 3900 nM T60529 CY65XB 10810622 IC50 = 30000 nM T60529 C68IWJ 10810738 IC50 > 100000 nM T60529 CLIV93 10810863 IC50 > 100000 nM T60529 CY4AX3 10811597 IC50 > 10000 nM T60529 C41MJH 10812437 IC50 = 3800 nM T60529 CQEP24 10812568 IC50 > 100000 nM T60529 COQ40E 10812673 IC50 > 100000 nM T60529 C30MWO 10812923 IC50 = 600 nM T60529 CPR41W 10816219 IC50 > 100000 nM T60529 C59HAF 10829130 IC50 = 33573.76 nM T60529 CZ0C4S 10829132 IC50 > 100000 nM T60529 CE92RY 10829314 IC50 = 2000 nM T60529 C50RZL 10830016 IC50 > 100000 nM T60529 CU6T5D 10830211 IC50 > 1000000 nM T60529 CG9A0R 10830212 IC50 > 100000 nM T60529 C3WOM2 10830272 IC50 = 6600 nM T60529 C2F1RB 10830394 IC50 = 10000 nM T60529 CKY2T4 10830950 IC50 = 2500 nM T60529 C7D4TN 10831290 IC50 = 16900 nM T60529 C56CIL 10831559 IC50 = 45800 nM T60529 CCLK02 10831725 IC50 = 770 nM T60529 CX97QO 10832104 IC50 = 27000 nM T60529 CMDL97 10832170 IC50 > 100000 nM T60529 CFXZ69 10832238 IC50 > 100000 nM T60529 CSCA58 10832407 IC50 > 100000 nM T60529 CJA96D 10832510 IC50 > 100000 nM T60529 C4JO1V 10832560 IC50 = 4500 nM T60529 CS2L9C 10833127 IC50 > 100000 nM T60529 CO8R6S 10833677 IC50 = 5794.29 nM T60529 CNE4F5 10834020 IC50 > 1000000 nM T60529 C54SBR 10834201 IC50 = 10900 nM T60529 C73TZG 10834744 IC50 > 100000 nM T60529 CE2HY4 10835226 IC50 > 100000 nM T60529 CUXE91 10835645 IC50 = 63600 nM T60529 CTU46J 10836128 IC50 = 38000 nM T60529 C6B8WX 10836221 IC50 > 100000 nM T60529 C12PJQ 10836527 IC50 = 35000 nM T60529 CHZW73 10850787 IC50 = 5000 nM T60529 CF98BX 10850793 IC50 = 200 nM T60529 C3PCB0 10851091 IC50 = 1500 nM T60529 C46JCP 10852345 IC50 = 150 nM T60529 CZI74A 10852952 IC50 > 100000 nM T60529 CIW26O 10853420 IC50 > 100000 nM T60529 CBVH56 10853804 IC50 > 100000 nM T60529 C9RQ7H 10854191 IC50 > 30000 nM T60529 C92EYG 10860016 IC50 = 5860 nM T60529 CLU6A5 10872407 IC50 > 1000 nM T60529 CWX81R 10872725 IC50 > 10000 nM T60529 C35PLX 10872752 IC50 > 10000 nM T60529 CB7IT1 10882387 IC50 > 10000 nM T60529 C1N4JQ 10882657 IC50 > 10000 nM T60529 C2JF4U 10882658 IC50 = 100000 nM T60529 C3DCA9 10893410 IC50 = 2700 nM T60529 C2S7FM 10893857 IC50 > 10000 nM T60529 CDHF71 10894407 IC50 > 10000 nM T60529 C1DQ9B 10901219 IC50 = 2640 nM T60529 CF0CX3 10904046 IC50 > 10000 nM T60529 C7DR3V 10908643 IC50 > 100 ug.mL-1 T60529 CJV6C1 10914501 IC50 > 10000 nM T60529 C5Y2AC 10914865 IC50 = 9880 nM T60529 COS6R7 10926603 IC50 > 10000 nM T60529 CAEI48 10936484 IC50 = 4700 nM T60529 CPNK84 10936619 IC50 > 100000 nM T60529 CP5W3G 10937079 IC50 = 47000 nM T60529 CYSJ65 10937794 IC50 = 4000 nM T60529 CD1N3J 10938268 IC50 > 1000 nM T60529 CTC5M0 10947004 IC50 > 100000 nM T60529 CSO6I1 10947517 IC50 > 100000 nM T60529 CTK81L 10948456 IC50 = 1300 nM T60529 CEA2N7 10960870 IC50 > 10000 nM T60529 C1K0DF 10980892 IC50 > 10000 nM T60529 C5VRD8 10981473 IC50 > 10000 nM T60529 C1RHL4 10990488 IC50 = 53 nM T60529 CT3PX2 10991144 IC50 = 480 nM T60529 C93BPL 10991235 IC50 = 5100 nM T60529 C9KIM8 10991648 IC50 > 10000 nM T60529 C74RTU 10991908 IC50 > 10000 nM T60529 C5FAQ4 10992868 IC50 > 10000 nM T60529 CY2J9R 11002614 IC50 > 100000 nM T60529 CS21NJ 11003065 IC50 = 29700 nM T60529 CQ3M8H 11012540 IC50 > 10000 nM T60529 C24SDE 11024492 IC50 > 10000 nM T60529 C0O4NS 11025223 IC50 > 10000 nM T60529 CQK2S8 11025447 IC50 > 10000 nM T60529 CGSD64 11034312 IC50 = 4100 nM T60529 CT2CH1 11035516 IC50 > 10000 nM T60529 CG4QE8 11036302 IC50 = 110 nM T60529 C5XQ9U 11036926 IC50 > 10000 nM T60529 C81NLC 11046361 IC50 > 10000 nM T60529 CMW94C 11046805 IC50 > 10000 nM T60529 C1O6JT 11046829 IC50 > 10000 nM T60529 C15YND 11056746 IC50 > 100000 nM T60529 CX60IR 11058879 IC50 > 10000 nM T60529 CY9UA1 11067599 IC50 > 10000 nM T60529 CE1V0L 11067992 IC50 > 10000 nM T60529 CW5F0A 11068088 IC50 = 40000 nM T60529 CQ8G6P 11068955 IC50 > 10000 nM T60529 CCM59W 11078663 IC50 = 3100 nM T60529 CP38KM 11079294 IC50 = 110 nM T60529 CTB97E 11079400 IC50 = 900 nM T60529 C37LKH 11089551 IC50 > 100000 nM T60529 CW13NO 11090142 IC50 > 10000 nM T60529 CHK0J7 11097158 IC50 = 5860 nM T60529 C5AD1I 11099739 IC50 > 100000 nM T60529 CW47TJ 11100014 IC50 > 10000 nM T60529 C75GDS 11110406 IC50 > 10000 nM T60529 CXP08O 11110905 IC50 > 10000 nM T60529 C31WGY 11112513 IC50 > 10000 nM T60529 CK57PL 11121068 IC50 > 10000 nM T60529 CC35GO 11122307 IC50 > 10000 nM T60529 CFSO12 11142523 IC50 > 10000 nM T60529 C3BJP2 11146784 IC50 > 100 ug.mL-1 T60529 C4P3WN 11150512 IC50 = 7440 nM T60529 CX0Q9R 11152069 IC50 = 1410 nM T60529 CXEA13 11154503 IC50 > 100000 nM T60529 C2AI8T 11155025 IC50 > 100000 nM T60529 CBRW71 11156027 IC50 = 36 nM T60529 CW1M8Q 11160272 IC50 = 13000 nM T60529 C3I1XG 11178642 IC50 = 6000 nM T60529 C7MY6G 11187835 IC50 = 39000 nM T60529 CC73ID 11196115 IC50 = 39000 nM T60529 C9J2CU 11196915 IC50 = 140 nM T60529 CU82SZ 11202736 IC50 = 17590 nM T60529 C8H4TN 11209828 IC50 = 410 nM T60529 C9JQK4 11211879 IC50 = 14000 nM T60529 CU01PR 11213050 IC50 > 100000 nM T60529 CM5Z6L 11213438 IC50 = 25050 nM T60529 CYX84A 11213988 IC50 = 38080 nM T60529 CDH1L4 11222461 IC50 > 10000 nM T60529 C5X0IY 11222615 IC50 > 100000 nM T60529 C5TBH9 11231244 IC50 > 100000 nM T60529 CC8Y0G 11234177 IC50 > 100000 nM T60529 CEX39T 11244379 IC50 = 7300 nM T60529 CP6N5B 11256540 IC50 = 260 nM T60529 C7EU3W 11256603 IC50 = 25610 nM T60529 CAT7H5 11257238 IC50 = 2910 nM T60529 CD0T4Y 11259519 IC50 = 44330 nM T60529 C6TQW2 11278070 IC50 = 140 nM T60529 C1HQ0V 11278404 IC50 = 2440 nM T60529 CTSE12 11279052 IC50 = 71100 nM T60529 C4SKT7 11279733 IC50 > 100000 nM T60529 C4TM3I 11280986 IC50 = 32000 nM T60529 C9EAJ5 11281693 IC50 > 100000 nM T60529 CY8K9F 11282341 IC50 > 100000 nM T60529 CA4S1X 11288276 IC50 = 1300 nM T60529 CAXV25 11291135 IC50 = 2270 nM T60529 CYR5J9 11292742 IC50 = 18800 nM T60529 C5M6EP 11301001 IC50 = 1030 nM T60529 CU3M8C 11301795 IC50 > 100000 nM T60529 C6NI5K 11301895 IC50 > 10000 nM T60529 C8ZGQ9 11302033 IC50 > 100000 nM T60529 C6L0BA 11302745 IC50 > 100000 nM T60529 CI6LW1 11313752 IC50 = 13200 nM T60529 C5BSC7 11316581 IC50 > 100000 nM T60529 C0NC7H 11317417 IC50 = 1560 nM T60529 CGL2N3 11336129 IC50 = 30000 nM T60529 CLR35D 11337592 IC50 = 25000 nM T60529 C8RH4F 11338802 IC50 = 37068.07 nM T60529 CTA54I 11340629 IC50 > 100000 nM T60529 C09HXJ 11340857 IC50 = 1810 nM T60529 COY06A 11359466 IC50 = 4630 nM T60529 CB8NC3 11361946 IC50 > 100000 nM T60529 CAQ0L4 11368202 IC50 = 51300 nM T60529 C2UG5L 11372471 IC50 > 40000 nM T60529 CL7X1Z 11373641 IC50 = 3790 nM T60529 C2EJ0X 11374699 IC50 > 100000 nM T60529 CF4JK1 11382191 IC50 > 100000 nM T60529 CDU98V 11382825 IC50 > 100000 nM T60529 C3F9SU 11382984 IC50 > 100000 nM T60529 CA85FN 11383735 IC50 = 207000 nM T60529 CR8T2S 11384636 IC50 = 13699.35 nM T60529 C3GOD4 11395292 IC50 = 3828 nM T60529 C1EL8Z 11396529 IC50 > 100000 nM T60529 CGQK95 11398561 IC50 = 25700 nM T60529 C1VYZ9 11404334 IC50 = 63900 nM T60529 C7DLM6 11405875 IC50 = 400 nM T60529 C02PEI 11415723 IC50 > 100000 nM T60529 C8LG9O 11416157 IC50 = 2300 nM T60529 CG9BL5 11417961 IC50 > 100000 nM T60529 CLC2X3 11418074 IC50 = 17200 nM T60529 C6JL8U 11419147 IC50 = 119000 nM T60529 C1ICK8 11430770 IC50 = 99560 nM T60529 C07IKF 11439406 IC50 > 100000 nM T60529 CDHJ18 11440364 IC50 = 3880 nM T60529 C4F9NZ 11440998 IC50 > 100000 nM T60529 CI6AL4 11442938 IC50 = 1130 nM T60529 C71AVE 11459907 IC50 > 10000 nM T60529 CR2WK3 11462316 IC50 = 270 nM T60529 CTAE25 11463338 IC50 > 100000 nM T60529 CSV5L3 11463339 IC50 = 1370 nM T60529 CQ7G3L 11464135 IC50 = 75900 nM T60529 C8P1SR 11472579 IC50 = 180 nM T60529 CB17JQ 11474778 IC50 > 100000 nM T60529 CFKU15 11483401 IC50 = 10860 nM T60529 CTFW72 11485547 IC50 > 100000 nM T60529 C6H1KP 11487377 IC50 > 100000 nM T60529 CD43NT 11487702 IC50 = 15810 nM T60529 CXU3T1 11487950 IC50 = 7140 nM T60529 CH0X2T 11500030 IC50 = 169000 nM T60529 C23SUC 11507797 IC50 = 30800 nM T60529 CO3ZL4 11544207 IC50 = 4200 nM T60529 C68AWO 11544686 IC50 = 173780.08 nM T60529 CKGE25 11544925 IC50 = 500 nM T60529 CY29OV 11546127 IC50 = 3300 nM T60529 C54ZXY 11552163 IC50 = 100000 nM T60529 C8DB6N 11609224 IC50 = 29800 nM T60529 C6FXD8 11649854 IC50 = 19900 nM T60529 CX0TY6 11688434 IC50 = 116 nM T60529 CIQ9A0 11693043 IC50 = 136000 nM T60529 CSQ1H3 11695155 IC50 = 3300 nM T60529 C03NOZ 11717695 IC50 = 141253.75 nM T60529 C5EX8K 11725274 IC50 = 6400 nM T60529 CQ8XW0 11725371 IC50 > 100000 nM T60529 CH2ZL7 11725645 IC50 = 12500 nM T60529 C2ONQ8 11726707 IC50 = 1500 nM T60529 C9BL0Q 11729490 IC50 > 10000 nM T60529 CP9N3Z 11731899 IC50 > 10000 nM T60529 CU8A0P 11731997 IC50 > 10000 nM T60529 CV7WN8 11731998 IC50 > 10000 nM T60529 CM4K3F 11732339 IC50 = 1900 nM T60529 C8CDF0 11739083 IC50 = 620 nM T60529 CK9H3A 11740421 IC50 = 105000 nM T60529 C65UAF 11744687 IC50 = 47000 nM T60529 CU28LA 11749849 IC50 = 240 nM T60529 C18WRI 11759902 IC50 > 10000 nM T60529 C69TMU 11759943 IC50 = 25000 nM T60529 C5XM3U 11760393 IC50 = 23800 nM T60529 C7CU9F 11761076 IC50 > 10000 nM T60529 C43QRI 11772569 IC50 = 360 nM T60529 C5YRB8 11774557 IC50 > 50000 nM T60529 CWLV48 11777274 IC50 > 100000 nM T60529 C8RG2P 11779569 IC50 = 45 nM T60529 C70YSD 11783741 IC50 > 10000 nM T60529 CDPH16 11791745 IC50 = 15000 nM T60529 CJRD74 11792200 IC50 = 35399.73 nM T60529 CPJA32 11792223 IC50 = 1750 nM T60529 C12XFM 11792433 IC50 > 100000 nM T60529 C3QOZ8 11792902 IC50 > 100000 nM T60529 C5MUO6 11793188 IC50 > 100000 nM T60529 C5HN3X 11793632 IC50 > 100000 nM T60529 C8UZS4 11793960 IC50 > 100000 nM T60529 C82BSG 11793963 IC50 > 100000 nM T60529 CPMF06 11794210 IC50 > 1000000 nM T60529 CW73EF 11794212 IC50 > 100000 nM T60529 CT29JD 11794221 IC50 > 10000 nM T60529 CUB83Z 11794411 IC50 > 100000 nM T60529 CKS37H 11794412 IC50 > 1000000 nM T60529 CZQU12 11795080 IC50 > 100000 nM T60529 CW96FD 11795129 IC50 > 100000 nM T60529 C8TI9K 11795549 IC50 > 100000 nM T60529 C3G8OL 11795928 IC50 > 100000 nM T60529 CO5Y9J 11795942 IC50 = 2100 nM T60529 C1YXB9 11796738 IC50 > 100000 nM T60529 C9O6SQ 11797537 IC50 > 100000 nM T60529 C8R7HN 11797837 IC50 > 1000000 nM T60529 CVT0F8 11808877 IC50 = 6900 nM T60529 CL28AI 11809792 IC50 = 1800 nM T60529 CQU0Z5 11810629 IC50 > 10000 nM T60529 CLW72J 11823443 IC50 = 61 nM T60529 CG9NH0 11823791 IC50 > 10000 nM T60529 C48YQU 11825301 IC50 > 10000 nM T60529 CK1F5U 11825947 IC50 > 10000 nM T60529 CXY1K6 11853318 IC50 > 100000 nM T60529 C0Y1KG 11853319 IC50 = 2400 nM T60529 CU9GT7 11853320 IC50 < 1000 nM T60529 CO2TH7 11853321 IC50 < 300 nM T60529 C8UG1W 11853323 IC50 > 10000 nM T60529 C6P4KS 11853563 IC50 = 3700 nM T60529 C1ZAM7 11853569 IC50 = 4700 nM T60529 CVO72K 11853818 IC50 > 100000 nM T60529 C06AVS 11853819 IC50 = 3600 nM T60529 CKHU91 11853820 IC50 < 1000 nM T60529 C8K3DI 11853821 IC50 = 15900 nM T60529 CT7A0W 11853822 IC50 = 2600 nM T60529 C7UIV6 11853823 IC50 = 1200 nM T60529 CO86TN 11854082 IC50 = 3000 nM T60529 CBW01R 11854339 IC50 = 1900 nM T60529 CG3WU6 11854340 IC50 = 11000 nM T60529 C2YRM5 11856982 IC50 = 5400 nM T60529 CEK42C 11856983 IC50 > 100000 nM T60529 CD68SB 11856984 IC50 = 1600 nM T60529 CS4XN1 11994185 IC50 > 50000 nM T60529 CV29NY 12015271 IC50 = 39700 nM T60529 C4GP2H 12080914 IC50 > 100000 nM T60529 CNE6W8 12088670 IC50 = 1800 nM T60529 C0U6WC 12130600 IC50 > 150000 nM T60529 CN8RP5 12306720 IC50 > 30000 nM T60529 CQL7T8 13148385 IC50 = 1900 nM T60529 CUAN95 13148390 IC50 > 25000 nM T60529 C0SZJ2 13148391 IC50 = 20200 nM T60529 CTH23W 13148392 IC50 = 4700 nM T60529 CHM37E 13148394 IC50 = 6300 nM T60529 C5L7XU 13148395 IC50 = 1300 nM T60529 CPE4D9 13609513 IC50 = 19000 nM T60529 C6BR7D 13609518 IC50 = 30000 nM T60529 CYK3G6 13804275 IC50 > 100000 nM T60529 CZQW71 13845711 IC50 = 18670 nM T60529 CM2NZ8 13986997 IC50 > 50000 nM T60529 CE0D3W 14015948 IC50 = 78000 nM T60529 C19KXV 14256046 IC50 = 10000 nM T60529 CS1XR2 14448070 IC50 > 200000 nM T60529 CS46EO 15153337 IC50 = 60 nM T60529 CKQ06L 15293126 IC50 = 13600 nM T60529 CY43FD 15340372 IC50 = 1000 nM T60529 C7KDB9 15345555 IC50 = 7100 nM T60529 C0MNT2 15345565 IC50 = 790 nM T60529 C9V0SW 15345568 IC50 = 299.99 nM T60529 CKB73V 15380222 IC50 > 100000 nM T60529 C7D5HB 15380227 IC50 > 100000 nM T60529 CXS52V 15388843 IC50 > 50000 nM T60529 CN4M6X 15388846 IC50 = 25000 nM T60529 C1WVD9 15388847 IC50 > 50000 nM T60529 CIV0Q3 15390770 IC50 = 5400 nM T60529 CR0QX1 15390771 IC50 = 230 nM T60529 CKOA87 15390773 IC50 > 100000 nM T60529 C7ZYU9 15406810 IC50 = 759.98 nM T60529 C20GFH 15428927 IC50 = 1300 nM T60529 CFP7D1 15429218 IC50 = 60000 nM T60529 C31OBS 15429221 IC50 > 100000 nM T60529 CFMC16 15429222 IC50 > 100000 nM T60529 C1WDE7 15429226 IC50 = 93000 nM T60529 CI93RK 15431535 IC50 > 10000 nM T60529 C0AFD5 15431540 IC50 > 10000 nM T60529 C57CWU 15431541 IC50 = 1000 nM T60529 CEK9A4 15453868 IC50 > 10000 nM T60529 C0F2NZ 15453869 IC50 > 10000 nM T60529 C90MOZ 15453870 IC50 = 10000 nM T60529 CB4R2G 15453871 IC50 = 490 nM T60529 CFZ3V5 15453872 IC50 = 120 nM T60529 CGQ15F 15453873 IC50 > 10000 nM T60529 C9I4JX 15461522 IC50 > 10000 nM T60529 C6OVQ9 15461525 IC50 = 3000 nM T60529 C8HE4A 15461526 IC50 > 100000 nM T60529 CUY31L 15461527 IC50 > 30000 nM T60529 C1W8LT 15485017 IC50 > 100000 nM T60529 CML5V6 15485782 IC50 = 1920 nM T60529 CV0W5O 15485784 IC50 = 1920 nM T60529 C1ZUI0 15516798 IC50 < 300 nM T60529 C3LIQ7 15516799 IC50 = 300 nM T60529 CT31VI 15516800 IC50 < 300 nM T60529 CYV58N 15521080 IC50 > 100000 nM T60529 C8PEQ1 15521081 IC50 = 30000 nM T60529 CC7J3Y 15524017 IC50 = 5800 nM T60529 C5C4IJ 15551252 IC50 > 1000000 nM T60529 CY2O8J 15551254 IC50 = 900 nM T60529 CYDT38 15617384 IC50 = 1100 nM T60529 C72QCS 15871000 IC50 = 600 nM T60529 CTS5M8 15871001 IC50 > 100000 nM T60529 C6LEP5 15887626 IC50 < 300 nM T60529 C2Z7BD 15887860 IC50 > 100000 nM T60529 CY31HD 15887862 IC50 = 83000 nM T60529 CTZN57 15887864 IC50 > 100000 nM T60529 CHT0D5 15887866 IC50 > 100000 nM T60529 CC09IL 15887878 IC50 = 39000 nM T60529 CH4RY6 16125421 IC50 > 100000 nM T60529 C0KTX5 16125422 IC50 > 100000 nM T60529 CH8PR5 16125423 IC50 > 100000 nM T60529 C86XQV 16125424 IC50 > 100000 nM T60529 C4P3AM 16125427 IC50 > 100000 nM T60529 CHR83T 16125428 IC50 > 100000 nM T60529 C8HKG4 16125488 IC50 > 100000 nM T60529 C1PC2X 16125489 IC50 > 100000 nM T60529 CX5WF4 16125491 IC50 > 100000 nM T60529 CE6J5R 16659826 IC50 > 400000 nM T60529 CHZ67I 16679964 IC50 > 33100 nM T60529 CMPG07 16679966 IC50 > 34900 nM T60529 C2DJ0O 16680045 IC50 > 33100 nM T60529 CU94BZ 16680046 IC50 > 34900 nM T60529 C4ZK0P 16730269 IC50 < 10000 nM T60529 CN8WX3 16757526 IC50 = 6700 nM T60529 CHX45B 16774693 IC50 > 100000 nM T60529 CPY46E 16774950 IC50 = 94000 nM T60529 COL01E 16777326 IC50 > 100000 nM T60529 CXPT85 17816126 IC50 > 100000 nM T60529 C82XZE 17816357 IC50 = 72500 nM T60529 C4NZB0 17828963 IC50 > 100000 nM T60529 C8VBA3 17876325 IC50 > 100000 nM T60529 CKX7R6 17876403 IC50 > 100000 nM T60529 C3IF4O 17880562 IC50 = 39000 nM T60529 C52AKR 17919591 IC50 > 10000 nM T60529 CB76TO 17919592 IC50 = 10000 nM T60529 CZAV04 17919601 IC50 = 10000 nM T60529 C5WHF9 17919602 IC50 = 1000 nM T60529 CZ3Y4S 17919604 IC50 > 10000 nM T60529 CN78MC 17919609 IC50 > 10000 nM T60529 CNA75S 18400189 IC50 = 2700 nM T60529 CME6G0 18400199 IC50 > 100000 nM T60529 CIB46D 18542198 IC50 = 1000 nM T60529 C32YUX 18542229 IC50 = 47000 nM T60529 COY2S1 18542237 IC50 = 65.9 nM T60529 CHW34K 18542252 IC50 > 10000 nM T60529 CM29WC 18542265 IC50 = 1510 nM T60529 CHN16W 18542282 IC50 > 100000 nM T60529 CS8JB4 18542341 IC50 = 3050 nM T60529 CWD09Y 18542351 IC50 > 10000 nM T60529 CR3MG9 18542368 IC50 = 21400 nM T60529 C2KQ6W 18543182 IC50 = 62000 nM T60529 CTL49C 18678268 IC50 > 100000 nM T60529 C1Q0ZN 18701559 IC50 > 100000 nM T60529 CW4V5S 18933706 IC50 = 830 nM T60529 CC85QH 18946587 IC50 > 50000 nM T60529 CWF4D0 18969710 IC50 = 370 nM T60529 CBQL15 18969715 IC50 = 120 nM T60529 C2L4QT 18969738 IC50 = 4400 nM T60529 CJ24BR 18969753 IC50 = 2000 nM T60529 C6U5AR 18969768 IC50 = 45000 nM T60529 C9ZGX8 19361705 IC50 = 10000 nM T60529 CP85SE 19426793 IC50 = 2100 nM T60529 CNFL01 19594572 IC50 = 41000 nM T60529 CP34MI 20115449 IC50 > 100000 nM T60529 CP5EU3 20117519 IC50 = 7200 nM T60529 CX36PZ 20402500 IC50 = 750 nM T60529 C19NOQ 20553328 IC50 = 540000 nM T60529 CTU20F 20658522 IC50 > 50000 nM T60529 CF7BY0 20658551 IC50 > 50000 nM T60529 CLX62I 20826014 IC50 = 780 nM T60529 C49YZM 20876816 IC50 = 229086.77 nM T60529 CRF1N2 21472741 IC50 > 100000 nM T60529 CGP84X 21472742 IC50 = 3000 nM T60529 CDJI26 21472746 IC50 > 100000 nM T60529 CF9A1O 21472747 IC50 = 14000 nM T60529 C8XH0M 21472750 IC50 = 10000 nM T60529 C7SMC9 21472751 IC50 > 100000 nM T60529 C19WHN 21472753 IC50 > 90000 nM T60529 C7D9QM 21472754 IC50 = 30000 nM T60529 C29VBS 21472759 IC50 > 300000 nM T60529 CK1XQ5 21548774 IC50 = 750 nM T60529 C24QKO 21596130 IC50 = 5900 nM T60529 CK49UX 21626480 IC50 > 50000 nM T60529 CUSW63 21626481 IC50 > 50000 nM T60529 CX8CM6 21630094 IC50 > 50000 nM T60529 CZUT41 21837604 IC50 = 350 nM T60529 CBS0C1 21858549 IC50 = 2800 nM T60529 CGC46S 21859783 IC50 = 810 nM T60529 CA1GV2 21859784 IC50 = 780 nM T60529 C1QV5P 21859785 IC50 = 700 nM T60529 C0VW7T 21859786 IC50 = 910 nM T60529 C4CQN5 21862750 IC50 = 60740 nM T60529 CI14XS 21883501 IC50 = 94200 nM T60529 C24DNQ 21883549 IC50 = 3110 nM T60529 C97AWR 21883555 IC50 < 350 nM T60529 CO12EU 21883567 IC50 = 140 nM T60529 C60ZGU 21883595 IC50 = 224000 nM T60529 COU74S 21883604 IC50 = 242 nM T60529 C3AQW5 21883607 IC50 = 3870 nM T60529 CRSU56 21883613 IC50 = 115000 nM T60529 CNW0V1 21883621 IC50 = 11000 nM T60529 CMY42K 21883631 IC50 = 33000 nM T60529 CVG02E 21948438 IC50 = 1000 nM T60529 C2FQO3 21948445 IC50 = 3000 nM T60529 C0HEC8 21948463 IC50 > 10000 nM T60529 CA09OG 21948479 IC50 > 10000 nM T60529 C41OLJ 21948498 IC50 = 3000 nM T60529 C2KU0M 21948499 IC50 > 10000 nM T60529 CF9E3P 21948521 IC50 = 300 nM T60529 CH7B4D 21948533 IC50 = 3000 nM T60529 C9I8LB 22034354 IC50 = 18000 nM T60529 CYAS85 22034360 IC50 = 33000 nM T60529 CLB58M 22034361 IC50 > 100000 nM T60529 CB2F0T 22034364 IC50 = 55700 nM T60529 CX6Q7U 22034367 IC50 = 12000 nM T60529 CMV2E3 22034374 IC50 = 18200 nM T60529 C3T6WH 22034376 IC50 = 33000 nM T60529 CZ2UB6 22034379 IC50 > 67000 nM T60529 CBDG24 22034386 IC50 = 8100 nM T60529 CF2N0H 22148957 IC50 > 50000 nM T60529 CVK2C0 22148978 IC50 = 49000 nM T60529 C08IZM 22562341 IC50 > 35100 nM T60529 CWRA65 22624559 IC50 > 100000 nM T60529 CO2X7W 22643554 IC50 > 100000 nM T60529 CF8M0T 22907695 IC50 = 3380 nM T60529 CNL89X 22911749 IC50 > 100000 nM T60529 CDOE75 22911767 IC50 > 100000 nM T60529 CM6HA9 22911810 IC50 = 19000 nM T60529 C3A4JD 22911832 IC50 > 10000 nM T60529 CHY0X9 22911835 IC50 = 120 nM T60529 C3U6GI 22911939 IC50 > 100000 nM T60529 CFID36 22911970 IC50 > 100000 nM T60529 CX5IO1 22911977 IC50 = 80 nM T60529 CT9Y7O 22911990 IC50 > 100000 nM T60529 CVOW97 22912028 IC50 > 100000 nM T60529 CI0C2S 22912091 IC50 > 100000 nM T60529 C9JP4B 22912100 IC50 > 10000 nM T60529 C0XL3N 22912115 IC50 > 100000 nM T60529 C0CT3B 22912123 IC50 > 100000 nM T60529 CBG45C 22912143 IC50 > 1000000 nM T60529 C8NS9E 22912151 IC50 > 100000 nM T60529 CX5B4Y 22912186 IC50 = 70000 nM T60529 CK4W3Z 22912196 IC50 > 1000000 nM T60529 C8GI4S 22912244 IC50 > 100000 nM T60529 C54EBF 22912306 IC50 > 100000 nM T60529 CW59QG 23002400 IC50 > 50000 nM T60529 CJYI21 23003613 IC50 = 849 nM T60529 CZV7D6 23225437 IC50 > 50000 nM T60529 CQ8O0J 23497471 IC50 > 100000 nM T60529 CC9PI3 23634884 IC50 = 20400 nM T60529 C62UXO 23663407 IC50 = 23500 nM T60529 CASU54 23696973 IC50 = 1258.93 nM T60529 C6UE8A 23717031 IC50 = 100000 nM T60529 CBXC05 24424330 IC50 = 8 nM T60529 C6DTY4 24689970 IC50 = 29000 nM T60529 CBR5L7 24695790 IC50 = 14000 nM T60529 CBU06J 24740875 IC50 < 300 nM T60529 COV92E 24752865 IC50 = 800 nM T60529 CELN62 24816405 IC50 = 87120 nM T60529 CD8PF6 24816406 IC50 > 100000 nM T60529 CUNJ72 24848656 IC50 = 660693.45 nM T60529 C4QEA8 24850953 IC50 = 96250 nM T60529 C85UXM 24853947 IC50 > 100000 nM T60529 C57ERS 24853948 IC50 > 100000 nM T60529 CP0DT5 24853949 IC50 = 12000 nM T60529 CV3ZL6 24853950 IC50 > 100000 nM T60529 CZ91QG 24854030 IC50 > 100000 nM T60529 CO8FU7 24854031 IC50 = 10000 nM T60529 C83WEO 24854032 IC50 > 100000 nM T60529 C4IP5C 24871714 IC50 = 62000 nM T60529 CE7TF2 24951013 IC50 = 86000 nM T60529 C69YHL 25000755 IC50 > 30000 nM T60529 CF1D8V 25028121 IC50 = 29700 nM T60529 CC9TW1 25034413 IC50 = 300 nM T60529 CWAR61 25072270 IC50 = 450 nM T60529 COMP96 25072271 IC50 = 600 nM T60529 CEFW12 25141402 IC50 = 21300 nM T60529 C3Y1RA 25188731 IC50 > 10000 nM T60529 CN8VX0 25188732 IC50 < 10000 nM T60529 CU1BY0 25188733 IC50 > 10000 nM T60529 CY30US 25188735 IC50 > 10000 nM T60529 CF64XU 25242322 IC50 = 11500 nM T60529 CHD71R 25242339 IC50 = 4100 nM T60529 CO83WB 25261943 IC50 = 2780 nM T60529 C8CWK5 42605184 IC50 = 4900 nM T60529 CXU63O 42607532 IC50 = 11700 nM T60529 CY19CJ 42609839 IC50 > 10000 nM T60529 C6DAY7 42609841 IC50 > 10000 nM T60529 C3SHI8 44138220 IC50 = 20000 nM T60529 C95VMW 44194809 IC50 = 1300 nM T60529 CR0ZJ5 44194810 IC50 = 7600 nM T60529 CCI14S 44194811 IC50 = 320 nM T60529 C4G7KU 44194812 IC50 = 1900 nM T60529 CE8B1R 44194813 IC50 = 1900 nM T60529 CJ8MZ9 44194814 IC50 = 810 nM T60529 CCZ52W 44194816 IC50 > 100000 nM T60529 C7NCJ3 44249752 IC50 = 720000 nM T60529 CR68BA 44250281 Ki > 25118.86 nM T60529 C8C7HF 44266438 IC50 > 100000 nM T60529 C7LT2W 44266451 IC50 > 100000 nM T60529 CC6W5I 44266508 IC50 > 100000 nM T60529 CGO38W 44269688 IC50 = 20000 nM T60529 C1W6AG 44271105 IC50 > 100000 nM T60529 CYHD60 44271141 IC50 > 100000 nM T60529 CP14AY 44271257 IC50 = 115000 nM T60529 C1ZT4X 44271312 IC50 = 1840 nM T60529 C0KMS2 44271350 IC50 = 10 nM T60529 CVC65J 44271374 IC50 = 4180 nM T60529 C9Q7AY 44271388 IC50 = 35600 nM T60529 CR18XW 44271618 IC50 = 730 nM T60529 C6HY3T 44271914 IC50 = 340 nM T60529 C3AQB6 44271916 IC50 = 1360 nM T60529 CD0G2T 44271975 IC50 = 570 nM T60529 C65LRW 44271985 IC50 = 250 nM T60529 CPFB09 44272072 IC50 > 100000 nM T60529 CT5JK3 44272073 IC50 > 100000 nM T60529 CAH19S 44272086 IC50 = 35000 nM T60529 CW1V9M 44272115 IC50 > 100000 nM T60529 CR97YP 44272129 IC50 > 10000 nM T60529 CCG76A 44272130 IC50 > 10000 nM T60529 CA12DG 44272131 IC50 = 7000 nM T60529 CVP23I 44272272 IC50 > 300000 nM T60529 C8M5HD 44272274 IC50 > 100000 nM T60529 C84VER 44272279 IC50 > 10000 nM T60529 C62UAH 44272281 IC50 = 81000 nM T60529 C59XIC 44272282 IC50 > 100000 nM T60529 CMDE94 44275919 IC50 = 15500000 nM T60529 CTC2U6 44286188 IC50 = 620 nM T60529 C74AXR 44286194 IC50 > 100000 nM T60529 C3DQM8 44286210 IC50 = 4900 nM T60529 C16ZON 44286326 IC50 ~ 100000 nM T60529 C7HM5U 44286327 IC50 = 9300 nM T60529 C1I7BA 44286343 IC50 = 12000 nM T60529 CYFP05 44286434 IC50 > 100000 nM T60529 CZ8YW9 44286540 IC50 = 6100 nM T60529 C0GH2Z 44286564 IC50 > 100000 nM T60529 C0D8JY 44289750 IC50 = 16700 nM T60529 C2PX9L 44292803 IC50 < 1240 nM T60529 CQ8VR4 44292819 IC50 > 100000 nM T60529 C5MCZ4 44292887 IC50 > 100000 nM T60529 CPM5C9 44293185 IC50 > 100000 nM T60529 CP16JH 44293186 IC50 = 29000 nM T60529 CPS6C2 44293290 IC50 > 100000 nM T60529 CNG5E2 44293477 IC50 = 9800 nM T60529 CN5FO1 44293478 IC50 = 5100 nM T60529 CNJ6W7 44293738 IC50 = 6900 nM T60529 C40VHQ 44293755 IC50 = 2400 nM T60529 CLJ6N1 44293775 IC50 = 2300 nM T60529 C0BM5Q 44293785 IC50 = 8200 nM T60529 CF7J1T 44293786 IC50 = 2500 nM T60529 CMG7L9 44293798 IC50 = 2700 nM T60529 C7SYX6 44293966 IC50 = 2680 nM T60529 CY4IZ3 44293967 IC50 = 7200 nM T60529 C9GIL0 44293982 IC50 = 5280 nM T60529 CB5ZI8 44293983 IC50 = 3700 nM T60529 C6BQR4 44293986 IC50 = 2500 nM T60529 CPH1M8 44294002 IC50 = 4000 nM T60529 CST64C 44294003 IC50 = 2500 nM T60529 C4YA8T 44307351 IC50 = 15000 nM T60529 CY4C8G 44307447 IC50 = 980 nM T60529 CN2YL4 44307454 IC50 > 50000 nM T60529 C0TCY3 44307455 IC50 > 50000 nM T60529 C3Y1FP 44307489 IC50 = 32000 nM T60529 CANV95 44307492 IC50 > 50000 nM T60529 CZ8QF9 44307510 IC50 > 50000 nM T60529 C7LH0E 44307511 IC50 = 750 nM T60529 CBRU60 44307554 IC50 = 17000 nM T60529 CU80YE 44307569 IC50 > 100000 nM T60529 CAT54L 44307599 IC50 > 50000 nM T60529 CYK0M4 44307760 IC50 = 3200 nM T60529 C82SQB 44316044 IC50 > 100000 nM T60529 CJ2A1Y 44316046 IC50 > 100000 nM T60529 C9K2HM 44316112 IC50 > 100000 nM T60529 CPUF05 44316113 IC50 = 490 nM T60529 CQVU84 44316126 IC50 > 100000 nM T60529 CA9W4P 44316373 IC50 = 7 nM T60529 CS8P4H 44323766 IC50 > 100000 nM T60529 CLN5J2 44323818 IC50 > 100000 nM T60529 CP4V8T 44323830 IC50 > 100000 nM T60529 CZ0RT7 44323831 IC50 > 100000 nM T60529 CK93EF 44324030 IC50 = 500 nM T60529 CL36JK 44325870 IC50 > 250000 nM T60529 CAU4X9 44325888 IC50 > 250000 nM T60529 C2KB1O 44326499 IC50 > 100000 nM T60529 CL6G5D 44326522 IC50 = 45000 nM T60529 CQ5HM8 44326892 IC50 = 6000 nM T60529 C74TXM 44326894 IC50 > 100000 nM T60529 CCF6N9 44327823 IC50 = 270 nM T60529 CYH73O 44327824 IC50 > 100000 nM T60529 CG95FW 44327825 IC50 > 100000 nM T60529 CBK0Y9 44327826 IC50 = 2670 nM T60529 C9XN8L 44327837 IC50 > 100000 nM T60529 CQF89I 44327838 IC50 = 11099.41 nM T60529 C52FEI 44327839 IC50 = 2730 nM T60529 CMHZ15 44327884 IC50 = 6240 nM T60529 C19PLO 44330414 IC50 = 10000 nM T60529 C9G4VJ 44330429 IC50 > 50000 nM T60529 CJ3CA1 44330646 IC50 > 100000 nM T60529 C78ANR 44338168 IC50 > 10000 nM T60529 C0TNX5 44338327 IC50 = 4600 nM T60529 C43QKL 44338544 IC50 = 1000 nM T60529 CV07XW 44343489 IC50 = 9000 nM T60529 C53XTU 44343803 IC50 = 600 nM T60529 C6IUT2 44343844 IC50 > 10000 nM T60529 CMKY74 44343870 IC50 = 10800 nM T60529 C5H0EO 44343879 IC50 > 100000 nM T60529 C4GM9U 44343958 IC50 > 10000 nM T60529 CR3F9L 44344532 IC50 = 20 nM T60529 CP6C3D 44344591 IC50 = 5000 nM T60529 C5OU6Q 44344842 IC50 = 75 nM T60529 C0QGP5 44344893 IC50 > 100000 nM T60529 C0KD4U 44346053 IC50 > 80000 nM T60529 CH0O5Q 44346322 IC50 > 80000 nM T60529 C2I4UH 44365341 IC50 > 50000 nM T60529 CN53LW 44365508 IC50 > 50000 nM T60529 CX64FE 44365531 IC50 > 50000 nM T60529 CA8RK2 44365569 IC50 > 50000 nM T60529 CBG3R5 44365570 IC50 > 50000 nM T60529 CKM4L8 44365743 IC50 = 320 nM T60529 CSVX52 44365745 IC50 = 78 nM T60529 CTWC52 44365758 IC50 > 50000 nM T60529 CP8MK0 44365764 IC50 > 50000 nM T60529 C67VZW 44366425 IC50 = 500 nM T60529 C26CIT 44366550 IC50 = 200 nM T60529 C8R1HW 44366732 IC50 = 3600 nM T60529 CCX61K 44366749 IC50 = 74 nM T60529 C2BSY4 44366835 IC50 = 1700 nM T60529 CAJ6R5 44366863 IC50 = 6400 nM T60529 CH84ZU 44366864 IC50 = 5400 nM T60529 CH35MX 44366879 IC50 = 6300 nM T60529 CLQ57F 44368274 IC50 > 1000000 nM T60529 CX8E3O 44368275 IC50 = 18400 nM T60529 CTJV50 44368294 IC50 = 1000000 nM T60529 CKO15H 44368313 IC50 = 229000 nM T60529 CE3O2K 44368376 IC50 = 56000 nM T60529 CH48YB 44368385 IC50 = 32400 nM T60529 CTCL75 44368677 IC50 > 1000000 nM T60529 CG9IE8 44370479 IC50 = 3000 nM T60529 C43QVB 44370496 IC50 = 10000 nM T60529 C6PQ8I 44370503 IC50 = 3000 nM T60529 CJUC35 44370506 IC50 = 10000 nM T60529 C8X3GE 44370516 IC50 > 10000 nM T60529 CER97H 44370520 IC50 = 10000 nM T60529 C1FZ8D 44370521 IC50 = 3000 nM T60529 CER2T7 44370528 IC50 > 10000 nM T60529 C2KAB9 44370560 IC50 = 10000 nM T60529 C61DTQ 44370597 IC50 > 10000 nM T60529 C8U0HS 44370604 IC50 > 10000 nM T60529 CZI0B6 44370618 IC50 = 10000 nM T60529 CM72JP 44370626 IC50 > 10000 nM T60529 CG4RK8 44370627 IC50 > 10000 nM T60529 CW21SL 44370636 IC50 > 10000 nM T60529 CFA7R3 44370649 IC50 = 10000 nM T60529 CV62SH 44370724 IC50 > 10000 nM T60529 CP3C8D 44370735 IC50 > 10000 nM T60529 C1JL9O 44370742 IC50 > 10000 nM T60529 CH9XR0 44370744 IC50 > 10000 nM T60529 C9JG2T 44370777 IC50 = 10000 nM T60529 C7EBG2 44370786 IC50 = 10000 nM T60529 C5M3UI 44370787 IC50 > 10000 nM T60529 CFB0R4 44370791 IC50 = 10000 nM T60529 C23EBS 44370949 IC50 = 10000 nM T60529 CO8F6L 44371320 IC50 > 50000 nM T60529 CZ6NB9 44371399 IC50 > 50000 nM T60529 CRKX10 44371400 IC50 > 50000 nM T60529 CG2LE1 44371407 IC50 > 50000 nM T60529 CNAY39 44371411 IC50 > 50000 nM T60529 CB1VP9 44371422 IC50 = 1100 nM T60529 CF9M7G 44371423 IC50 > 50000 nM T60529 CU87HG 44371424 IC50 = 610 nM T60529 C4EH5S 44371430 IC50 = 8500 nM T60529 C0GSH9 44371442 IC50 = 9000 nM T60529 CZY89I 44371457 IC50 > 50000 nM T60529 CV5CT2 44371478 IC50 = 30000 nM T60529 CJ1B2O 44371479 IC50 = 15000 nM T60529 C09UKQ 44371492 IC50 = 9600 nM T60529 C58UDX 44371493 IC50 = 600 nM T60529 CL2SU4 44371522 IC50 = 2400 nM T60529 CNBA18 44373038 IC50 > 500000 nM T60529 CM3JR7 44373310 IC50 > 500000 nM T60529 CT03QD 44373312 IC50 > 500000 nM T60529 C5UC8Z 44373338 IC50 > 500000 nM T60529 CSB9D6 44373350 IC50 > 500000 nM T60529 CL85CK 44373654 IC50 > 500000 nM T60529 C2IY7Z 44374212 IC50 > 100000 nM T60529 CO0Q1M 44374403 IC50 > 100000 nM T60529 C65YTP 44375433 IC50 = 34400 nM T60529 CKW4V5 44375673 IC50 = 9400 nM T60529 CSPX90 44375691 IC50 = 2800 nM T60529 CXMA02 44378192 IC50 = 1300 nM T60529 C84GOY 44378193 IC50 > 10000 nM T60529 CH3J8M 44378194 IC50 > 10000 nM T60529 CG0L4N 44378225 IC50 = 38000 nM T60529 CKI2Y8 44382878 IC50 > 50000 nM T60529 C18EVN 44382879 IC50 > 100000 nM T60529 CV14NG 44383162 IC50 > 50000 nM T60529 C1QJ0T 44383441 IC50 > 50000 nM T60529 CG6YA9 44383560 IC50 > 50000 nM T60529 CG89SY 44383610 IC50 > 50000 nM T60529 C7DT4Q 44383772 IC50 > 50000 nM T60529 C59OQY 44383922 IC50 > 50000 nM T60529 C8D4RP 44384088 IC50 > 50000 nM T60529 C8M7RO 44387158 IC50 > 10000 nM T60529 C9A4FM 44393815 IC50 = 2440 nM T60529 CCDH14 44393845 IC50 = 6000 nM T60529 CO2RG9 44393852 IC50 = 6000 nM T60529 C37BAX 44393874 IC50 = 3500 nM T60529 CI9P5S 44393917 IC50 > 40000 nM T60529 C0FH8A 44393943 IC50 = 9300 nM T60529 CJA59H 44394041 IC50 = 16982.44 nM T60529 C0RU8B 44394065 IC50 = 1698.24 nM T60529 C80QPC 44394101 IC50 = 16595.87 nM T60529 C0LO6A 44394134 IC50 = 3890.45 nM T60529 C2UE8J 44394151 IC50 = 14791.08 nM T60529 CAC41P 44394156 IC50 = 17782.79 nM T60529 CW6PL2 44394178 IC50 = 588.84 nM T60529 CI3W1R 44394196 IC50 = 3715.35 nM T60529 CE0MN4 44394205 IC50 = 10964.78 nM T60529 CLO09F 44394229 IC50 = 5495.41 nM T60529 CK87TF 44394245 IC50 = 19054.61 nM T60529 CR3HM1 44394264 IC50 = 5754.4 nM T60529 CD5K3W 44394272 IC50 = 22387.21 nM T60529 CAH37E 44395024 IC50 > 100000 nM T60529 CTWD42 44395063 IC50 > 100000 nM T60529 CE1O8I 44395070 IC50 = 24100 nM T60529 C6GB9N 44395090 IC50 > 100000 nM T60529 C5IJZ0 44395098 IC50 > 19100 nM T60529 CYRL43 44395118 IC50 > 100000 nM T60529 CK1CQ3 44395128 IC50 = 2605 nM T60529 CM1C6S 44395142 IC50 = 8630 nM T60529 CA58EW 44395152 IC50 > 100000 nM T60529 C8V1IN 44395167 IC50 = 43900 nM T60529 C60XRQ 44395168 IC50 > 100000 nM T60529 CR9B7F 44395179 IC50 = 58300 nM T60529 CG1JZ6 44395210 IC50 > 100000 nM T60529 CH8KP6 44395250 IC50 > 100000 nM T60529 C74OSX 44400364 IC50 = 132000 nM T60529 CW89YC 44402559 IC50 > 8600 nM T60529 C5AVD1 44406245 IC50 > 100000 nM T60529 CC58ZJ 44406275 IC50 > 25000 nM T60529 CYJ4L1 44406281 IC50 = 285000 nM T60529 CN4JP6 44406313 IC50 = 105000 nM T60529 C5AIR7 44406314 IC50 = 62300 nM T60529 CH58AJ 44406315 IC50 > 100000 nM T60529 C7CBT6 44407538 IC50 = 38500 nM T60529 C62WEY 44407539 IC50 = 43000 nM T60529 C47PDJ 44407681 IC50 = 14400 nM T60529 CV2PF1 44407684 IC50 = 31300 nM T60529 CHS1Y0 44407685 IC50 = 48500 nM T60529 CX3CO6 44407686 IC50 = 221300 nM T60529 C2X5NT 44407723 IC50 = 18900 nM T60529 C2RCH3 44407952 IC50 = 19700 nM T60529 CEK62L 44407953 IC50 = 15700 nM T60529 CJW4T6 44407958 IC50 = 35500 nM T60529 CF50IJ 44408022 IC50 > 150000 nM T60529 CH87VZ 44415454 IC50 = 35070 nM T60529 C6L1HD 44415455 IC50 = 26260 nM T60529 CM37ED 44424015 IC50 < 10000 nM T60529 C6UM5Y 44424016 IC50 < 10000 nM T60529 C7K8UC 44431346 IC50 = 4700 nM T60529 CYBP49 44434498 IC50 = 1900 nM T60529 C59WCO 44435729 IC50 < 1000 nM T60529 CUPI01 44443328 IC50 = 53900 nM T60529 CC04HF 44443330 IC50 > 100000 nM T60529 CY5BC2 44447992 IC50 > 1000 nM T60529 C7UR1D 44447993 IC50 = 7700 nM T60529 C3V5BJ 44456558 IC50 = 23990 nM T60529 CRU0P2 44456559 IC50 = 56730 nM T60529 C9QMH1 44456607 IC50 = 31270 nM T60529 CH3BO6 44456631 IC50 = 51830 nM T60529 CIHG87 44456655 IC50 = 43890 nM T60529 CH89VO 44456656 IC50 = 64420 nM T60529 CS4J0Y 44473488 IC50 = 20020 nM T60529 CNW37Q 44473489 IC50 = 2120 nM T60529 CD0AT5 44473490 IC50 = 560 nM T60529 CD30GC 44473491 IC50 = 1310 nM T60529 CZ4C8E 44473492 IC50 = 3790 nM T60529 C2A4KE 44473493 IC50 = 2730 nM T60529 CPN75T 44473494 IC50 = 25240 nM T60529 C0MK9H 44473495 IC50 = 2060 nM T60529 C1AIL9 44473650 IC50 = 1150 nM T60529 CUE30M 44473651 IC50 = 8550 nM T60529 C6J2RO 44473652 IC50 = 270 nM T60529 CMV3R2 44473653 IC50 = 940 nM T60529 CUW67Z 44474131 IC50 = 190 nM T60529 CO92ZS 44474132 IC50 = 1090 nM T60529 CB25PR 44474133 IC50 = 1150 nM T60529 CI37VD 44474262 IC50 = 420 nM T60529 C0FX4E 44474277 IC50 = 910 nM T60529 CJ9GH7 44474278 IC50 = 1600 nM T60529 CUPE26 44474279 IC50 = 480 nM T60529 C4JO6Z 44474280 IC50 = 990 nM T60529 CCKA05 44474281 IC50 = 170 nM T60529 CS20YU 44474282 IC50 = 3250 nM T60529 CF34OX 44474283 IC50 = 690 nM T60529 C54TCU 44474284 IC50 = 1220 nM T60529 C5W2HM 44475682 IC50 = 2570 nM T60529 C58AIG 44475683 IC50 = 60390 nM T60529 CSEV14 44475684 IC50 = 9760 nM T60529 C7LM9A 44475685 IC50 = 560 nM T60529 CJG1Z8 44475687 IC50 = 80 nM T60529 C1MKA9 44475839 IC50 = 760 nM T60529 CXZ6M4 44475840 IC50 = 1110 nM T60529 CN20QC 44475841 IC50 = 1000 nM T60529 C3KSY1 44475842 IC50 = 100 nM T60529 C2JL7C 44475844 IC50 = 480 nM T60529 CFA7N0 44475845 IC50 = 7150 nM T60529 C52LKE 44475846 IC50 = 1310 nM T60529 C30XPZ 44541795 IC50 = 1.23 nM T60529 C35GON 44559963 IC50 = 42000 nM T60529 CM7N8F 44563734 IC50 = 12400 nM T60529 C3C9PD 44563736 IC50 = 11400 nM T60529 CJMV72 44563737 IC50 = 5300 nM T60529 C18NSI 44563762 IC50 = 290 nM T60529 CGP5B1 44563765 IC50 = 3200 nM T60529 CQ50LO 44563767 IC50 = 1900 nM T60529 CJE82G 44563770 IC50 = 4900 nM T60529 CND7B3 44563771 IC50 = 970 nM T60529 C0P7CV 44563772 IC50 = 32600 nM T60529 CGT24V 44563774 IC50 = 7800 nM T60529 CY24ED 44563802 IC50 = 16500 nM T60529 CJ48ZX 44563803 IC50 = 18400 nM T60529 CWP6H3 44563804 IC50 = 17800 nM T60529 C04FCZ 44563805 IC50 = 36300 nM T60529 CTB3C7 44563806 IC50 = 1900 nM T60529 CC71OE 44563807 IC50 = 10600 nM T60529 C84WIE 44563808 IC50 = 10500 nM T60529 CH3C5K 44563809 IC50 = 10900 nM T60529 C61AIS 44563811 IC50 = 10700 nM T60529 CHNO16 44563812 IC50 = 3000 nM T60529 C4B5RC 44563815 IC50 = 9700 nM T60529 C4X7MK 44563816 IC50 = 5400 nM T60529 C13MLD 44563817 IC50 = 990 nM T60529 CRT8Q1 44571459 IC50 = 7400 nM T60529 CJ5QM1 44571461 IC50 = 11600 nM T60529 C2A7RC 44571462 IC50 = 3500 nM T60529 CXZ1U2 44571463 IC50 = 170 nM T60529 CDL15O 44571464 IC50 = 30500 nM T60529 CXE3G5 44581926 IC50 = 20800 nM T60529 C82KLY 44581927 IC50 = 45000 nM T60529 CN0RZ4 44581928 IC50 = 10000 nM T60529 C48XMK 44581929 IC50 > 100000 nM T60529 C41WAT 44581930 IC50 = 12200 nM T60529 CN01BJ 44581931 IC50 = 12500 nM T60529 CU9R8L 44581948 IC50 = 830 nM T60529 CGWQ85 44581949 IC50 = 840 nM T60529 CVA10P 44582812 IC50 = 1000000 nM T60529 CA04YB 44582833 IC50 > 1000000 nM T60529 CE8QI7 44584103 IC50 > 100 ug.mL-1 T60529 C5GOW9 44584170 IC50 = 8300 nM T60529 C3S7OL 44584247 IC50 = 73000 nM T60529 CSFK23 44584256 IC50 = 64000 nM T60529 CT5J7E 44584264 IC50 = 40000 nM T60529 CE32JQ 44584275 IC50 = 43000 nM T60529 C25YEN 44584287 IC50 = 50000 nM T60529 CB96SQ 44584307 IC50 = 81000 nM T60529 CKV1H6 44584314 IC50 = 1000000 nM T60529 CLP0D9 44587062 IC50 = 17000 nM T60529 CD2G5H 44587408 IC50 = 580 nM T60529 CO28GQ 44587409 IC50 = 570 nM T60529 C3WRM5 44587410 IC50 = 480 nM T60529 C09XWJ 44587411 IC50 = 110000 nM T60529 CASI69 44587478 IC50 = 580 nM T60529 C1JKZ3 44587479 IC50 = 123000 nM T60529 CX54EY 44818111 IC50 = 24000 nM T60529 CZ31PF 45267710 IC50 = 100000 nM T60529 CV4YK9 45267715 IC50 = 6321 nM T60529 C9MC8Z 45267716 IC50 > 100000 nM T60529 C9TV1Z 45267717 IC50 > 100000 nM T60529 C3WXL0 45267733 IC50 > 52124 nM T60529 CNS9Z2 45267769 IC50 > 100000 nM T60529 C1BRY0 45267770 IC50 > 65800 nM T60529 CNW5D2 45268615 IC50 > 100000 nM T60529 CD2K4X 45268625 IC50 > 100000 nM T60529 CNP20Q 45268649 IC50 > 100000 nM T60529 C2EUZ7 45269433 IC50 > 74175 nM T60529 C2CBS0 45269451 IC50 = 1921 nM T60529 CU46BW 45269475 IC50 > 100000 nM T60529 CHU45M 45269513 IC50 = 167 nM T60529 C2KAY8 45270280 IC50 > 100000 nM T60529 C09BLU 45270285 IC50 = 52556 nM T60529 C8KT1R 45270290 IC50 = 4038 nM T60529 C5KMT9 45270336 IC50 > 100000 nM T60529 C8ETI0 45270348 IC50 > 96150 nM T60529 CMY4J7 45270349 IC50 = 700 nM T60529 CI18ZS 45271088 IC50 > 100000 nM T60529 CS07LK 45271115 IC50 = 3000 nM T60529 C6NPR3 45271129 IC50 > 100000 nM T60529 CZU07P 45271135 IC50 = 2969 nM T60529 CIR3V5 45271980 IC50 > 100000 nM T60529 C4BVM8 45271990 IC50 > 100000 nM T60529 CCBV52 45271997 IC50 = 52000 nM T60529 CXTE06 45271998 IC50 = 4357 nM T60529 C5AZ2N 45272015 IC50 > 100000 nM T60529 C6D0RE 45272025 IC50 = 6541 nM T60529 CLNJ85 45272026 IC50 = 29371 nM T60529 CY82CH 45272817 IC50 > 100000 nM T60529 C7RT6N 45272818 IC50 > 100000 nM T60529 CA6N3E 45272824 IC50 = 19000 nM T60529 CMU54J 45272831 IC50 > 34000 nM T60529 CR0FZ9 45272838 IC50 = 10000 nM T60529 C50WBE 45272855 IC50 > 100000 nM T60529 CJO71V 45273765 IC50 > 100000 nM T60529 C0E4AV 45273799 IC50 > 100000 nM T60529 CZ6YD5 45273803 IC50 = 4340 nM T60529 CF4C0H 45273829 IC50 > 100000 nM T60529 CJX28F 46213934 IC50 = 2500 nM T60529 CQRN43 46229713 IC50 = 125000 nM T60529 C8PZU1 46235580 IC50 = 25000 nM T60529 CE9CY1 46701619 IC50 = 12300 nM T60529 C6RV7G 46701878 IC50 > 10000 nM T60529 C9DRL8 46845033 IC50 = 7400 nM T60529 CRQ29W 46880352 IC50 > 50000 nM T60529 CYPD43 46892801 IC50 > 400000 nM T60529 C8MXU2 46906688 IC50 = 6000 nM T60529 C2KJ1L 46906728 IC50 = 24400 nM T60529 CFL89P 46906732 IC50 = 18200 nM T60529 CZ1BI2 46906736 IC50 = 7800 nM T60529 CDY1P0 46906738 IC50 = 36700 nM T60529 CT39AY 46906740 IC50 = 16500 nM T60529 CH1ZW7 46906744 IC50 = 180300 nM T60529 CO62DT 46906746 IC50 = 24000 nM T60529 CAT0M6 46926545 IC50 = 2 nM T60529 C2PL3G 46927848 IC50 > 10000 nM T60529 CI8P0A 46937277 IC50 > 1000000 nM T60529 CP03KU 49799224 IC50 = 7800 nM T60529 C0A2SK 49799225 IC50 = 6300 nM T60529 CV0SD4 49799226 IC50 = 8800 nM T60529 C9JL4Z 49799227 IC50 = 8900 nM T60529 CWYT40 49799228 IC50 = 7800 nM T60529 C8IP0B 49799229 IC50 = 7500 nM T60529 C1RA6K 49799230 IC50 = 8000 nM T60529 CU40RO 49799231 IC50 = 7600 nM T60529 CNR7J1 49799265 IC50 = 8800 nM T60529 CS4D9W 49799266 IC50 = 8300 nM T60529 CMS46L 49799267 IC50 = 5900 nM T60529 CBNJ36 49799268 IC50 > 50000 nM T60529 CZ28MX 49799269 IC50 > 50000 nM T60529 CBWS90 49799270 IC50 > 50000 nM T60529 C9L3UH 49799271 IC50 > 50000 nM T60529 CJQ4I0 49799272 IC50 > 50000 nM T60529 C0S2VP 49799273 IC50 > 50000 nM T60529 C78XZV 49804917 IC50 = 61000 nM T60529 CEHY29 49804918 IC50 > 100000 nM T60529 C6IWU7 49804919 IC50 = 20400 nM T60529 C8W3GR 49804920 IC50 > 100000 nM T60529 CQO37H 49805049 IC50 > 100000 nM T60529 CQD83P 49805050 IC50 > 100000 nM T60529 CC51BP 49805051 IC50 > 100000 nM T60529 C5L4CW 49805052 IC50 > 100000 nM T60529 C8JVU3 49805053 IC50 > 100000 nM T60529 C8XY3D 49805054 IC50 > 100000 nM T60529 C5MDK8 49805055 IC50 > 100000 nM T60529 C51KQC 49805174 IC50 > 100000 nM T60529 C8CER6 49805175 IC50 > 100000 nM T60529 C1LGX6 49805176 IC50 > 100000 nM T60529 C0HTK6 49805177 IC50 > 100000 nM T60529 CX6K0C 49805178 IC50 > 100000 nM T60529 C0S4FY 49805179 IC50 > 100000 nM T60529 CD8J0L 49805180 IC50 > 100000 nM T60529 CBK9A7 49805302 IC50 > 100000 nM T60529 CVD4T1 49805303 IC50 = 1900 nM T60529 CU34WJ 49805304 IC50 > 100000 nM T60529 CVI2E6 49805305 IC50 > 100000 nM T60529 CRV4K9 49805306 IC50 > 100000 nM T60529 CLR02I 49805307 IC50 > 100000 nM T60529 CG7EJ4 49837500 IC50 = 30000 nM T60529 CZ9UD6 50901657 IC50 > 100000 nM T60529 C4M2NP 50908173 IC50 = 96220 nM T60529 CUK21S 50908400 IC50 > 100000 nM T60529 CNHJ51 50908401 IC50 > 100000 nM T60529 C7AL4X 51003554 IC50 = 26500 nM T60529 C03UJK 51003555 IC50 = 24700 nM T60529 COX20E 51003556 IC50 > 100000 nM T60529 CU7ST1 51346826 IC50 > 100000 nM T60529 CMG36K 52826130 IC50 = 7210 nM T60529 CL6VB4 52826143 IC50 = 8320 nM T60529 CF6X5T 52826146 IC50 = 9200 nM T60529 CCG7T3 52918139 IC50 = 22870 nM T60529 C17IAT 52918154 IC50 = 14380 nM T60529 CSBE15 52918155 IC50 = 17170 nM T60529 C4Y9MC 52918156 IC50 = 19750 nM T60529 C26WPM 52941067 IC50 = 7700 nM T60529 C1OEI4 52941415 IC50 = 7000 nM T60529 CW5U1X 52941672 IC50 = 2200 nM T60529 CT4D1X 52942295 IC50 = 6300 nM T60529 CJFR43 52942521 IC50 = 1740 nM T60529 CR47KD 52942604 IC50 = 140 nM T60529 CV27HX 52942642 IC50 = 320 nM T60529 C9OED7 52942694 IC50 = 62700 nM T60529 C2Y5DB 52942695 IC50 = 2690 nM T60529 C0XOH5 52943192 IC50 = 9620 nM T60529 CZC8Q3 52943858 IC50 = 71700 nM T60529 CK52YW 52944376 IC50 = 4990 nM T60529 CM6CJ2 52946158 IC50 = 410 nM T60529 CQ5X9F 52946285 IC50 = 100000 nM T60529 C4K6BH 52946883 Ki > 100000 nM T60529 CBM7U1 52946890 IC50 = 2580 nM T60529 CZCN58 52948356 IC50 = 600 nM T60529 CQD5M1 52948912 IC50 = 100000 nM T60529 C0TXV9 52949921 IC50 = 120 nM T60529 CI9BQ4 52950184 IC50 = 7200 nM T60529 C3UEM7 53248884 IC50 = 326000 nM T60529 C1SA2Z 53249089 IC50 > 400000 nM T60529 C06YVC 53316515 IC50 > 100000 nM T60529 CKD6L2 53316516 IC50 = 740 nM T60529 C61HIM 53316646 IC50 = 440 nM T60529 C26NMZ 53317589 IC50 = 22600 nM T60529 CKT7G2 53317947 IC50 = 15800 nM T60529 CYJT73 53318566 IC50 = 38280 nM T60529 CK6NI5 53318567 IC50 = 29320 nM T60529 CQ0Z3T 53319059 IC50 = 100000 nM T60529 CA6H8Q 53319286 IC50 = 370 nM T60529 CRM4A0 53319287 IC50 = 100000 nM T60529 C3AD1U 53319288 IC50 = 3660 nM T60529 CTL23B 53320186 IC50 = 100000 nM T60529 CRIX73 53320474 IC50 > 100000 nM T60529 C2TO9G 53320589 IC50 < 140 nM T60529 CYJ7F1 53320590 IC50 = 41600 nM T60529 CX2WV0 53321196 IC50 = 21570 nM T60529 C6EO8G 53321885 IC50 = 48900 nM T60529 CVB21L 53321886 IC50 = 100000 nM T60529 CUTF34 53322523 IC50 = 22300 nM T60529 CE14JM 53322743 IC50 = 1390 nM T60529 C0GAC7 53323100 IC50 = 2440 nM T60529 CVUN53 53323101 IC50 = 4340 nM T60529 CUF68R 53323225 IC50 > 100000 nM T60529 CKL68J 53323226 IC50 = 100000 nM T60529 CY36BC 53323227 IC50 = 350 nM T60529 CM4L0D 53323860 IC50 = 26040 nM T60529 CQ5UV6 53324322 IC50 = 39800 nM T60529 CFTY39 53324454 IC50 = 17700 nM T60529 CHX7F1 53324576 IC50 > 100000 nM T60529 C9NE3C 53324577 IC50 = 1950 nM T60529 CXHQ58 53324578 IC50 = 1630 nM T60529 CN86CK 53325524 IC50 = 68400 nM T60529 CL37DN 53325623 IC50 = 27180 nM T60529 C68WVL 53325872 IC50 = 100000 nM T60529 C7HSA5 53325873 IC50 = 100000 nM T60529 CZ70LU 53326920 IC50 = 66700 nM T60529 C4U5IX 53493001 IC50 = 35000 nM T60529 CZJY42 54669869 IC50 = 9600 nM T60529 C6UAZ5 54669874 IC50 = 12200 nM T60529 COZ9N1 54685766 IC50 > 100 ug.mL-1 T60529 CEK6X8 54686705 IC50 = 6760 nM T60529 CGWP10 54690323 IC50 = 218 ug.mL-1 T60529 C4O1PT 54698884 IC50 = 19800 nM T60529 C87GPY 54728405 IC50 = 489000 nM T60529 C3IXM4 54728414 IC50 = 118000 nM T60529 C5GRB6 54754354 IC50 = 300 nM T60529 C3YM2E 54754518 IC50 > 10000 nM T60529 C6R9ES 54764159 IC50 = 35600 nM T60529 C79DVG 56589615 IC50 > 10000 nM T60529 CN3F5O 56641761 IC50 > 10000 nM T60529 C7ZI3H 56642018 IC50 > 10000 nM T60529 CU1G5A 56642290 IC50 = 41 nM T60529 C0SM7Z 56642536 IC50 = 900 nM T60529 C6TLW3 56642537 IC50 = 14 nM T60529 C4RC3Y 56661768 IC50 = 49000 nM T60529 C1MIO4 56665210 IC50 = 54000 nM T60529 CU2HX5 56665212 IC50 = 56000 nM T60529 CJMI28 56665214 IC50 > 1000000 nM T60529 CX30HR 56665216 IC50 = 310000 nM T60529 C5QZK1 56668661 IC50 = 515000 nM T60529 CHC69U 56668662 IC50 = 4000 nM T60529 CHS43U 56668663 IC50 = 270000 nM T60529 CFI7A8 56668664 IC50 = 93000 nM T60529 CS79OK 56668666 IC50 = 800000 nM T60529 C9QLO1 56668668 IC50 = 174000 nM T60529 C60GOL 56668670 IC50 = 470000 nM T60529 CPY6S5 56668671 IC50 = 47000 nM T60529 C47KYI 56672141 IC50 > 1000000 nM T60529 C7JEP3 56672143 IC50 = 575000 nM T60529 CCW0G2 56672144 IC50 = 174000 nM T60529 CM3X4L 56672145 IC50 > 1000000 nM T60529 CHX16S 56675533 IC50 = 460000 nM T60529 C23DNE 56675535 IC50 = 74000 nM T60529 CE74XR 56682184 IC50 = 758000 nM T60529 CI7AU6 56682186 IC50 = 650000 nM T60529 CC73ZT 56850255 IC50 = 18000 nM T60529 C2XBJ9 56850523 IC50 = 620 nM T60529 CK0I6Q 56850525 IC50 > 30000 nM T60529 CLJA61 56850666 IC50 = 3200 nM T60529 C4ZS8Q 56850668 IC50 = 9000 nM T60529 CRB5G2 56929489 IC50 = 600 nM T60529 CS1J6W 56929588 IC50 = 31240 nM T60529 CU6QX9 56929591 IC50 = 20000 nM T60529 CMUW75 56964580 IC50 = 495 nM T60529 C4O3HY 57391146 IC50 = 29800 nM T60529 CJCD09 57391147 IC50 = 41500 nM T60529 CX5CY1 57392459 IC50 = 54 nM T60529 CC2AF6 57392917 IC50 = 35800 nM T60529 C27JKX 57392918 IC50 = 42500 nM T60529 CU4OY7 57392919 IC50 > 50000 nM T60529 C5RP6B 57392920 IC50 = 43800 nM T60529 C76TYD 57393522 IC50 > 400000 nM T60529 CXI23L 57394660 IC50 = 35800 nM T60529 C2P6NT 57396409 IC50 > 50000 nM T60529 CM5J7X 57396410 IC50 = 40300 nM T60529 CWAI02 57396427 IC50 > 10000 nM T60529 C2GJQ6 57399859 IC50 > 50000 nM T60529 CSEF30 57399860 IC50 = 40200 nM T60529 CV1K0D 57401637 IC50 = 40500 nM T60529 C2LK4N 57401638 IC50 = 38000 nM T60529 CZV54H 57401639 IC50 > 50000 nM T60529 C0VB8K 57401640 IC50 = 39800 nM T60529 CM0YK9 57401647 IC50 > 10000 nM T60529 C20JKE 57403365 IC50 = 36900 nM T60529 CXCJ10 57403366 IC50 = 41200 nM T60529 CX9P8K 57563344 IC50 = 100000 nM T60529 C8J5WL 57780764 IC50 = 19200 nM T60529 CJK1Y2 57780765 IC50 > 100000 nM T60529 CXY02N 57780766 IC50 = 5000 nM T60529 CWXK91 57780767 IC50 = 4200 nM T60529 C37LRH 57780770 IC50 > 100000 nM T60529 CBUG72 57780771 IC50 = 2200 nM T60529 C9JQL6 57780772 IC50 > 100000 nM T60529 CEYZ93 57780773 IC50 = 270 nM T60529 C02TNX 57780777 IC50 > 100000 nM T60529 CK0RX3 57780779 IC50 = 17400 nM T60529 C21WOV 58934890 IC50 > 100000 nM T60529 CXLV30 60155351 IC50 = 1500 nM T60529 CP5O0C 60155353 IC50 = 3000 nM T60529 CG68SH 60155450 IC50 = 9000 nM T60529 CS4Q0U 60155529 IC50 = 15600 nM T60529 CEU8V0 60155531 IC50 = 21600 nM T60529 CGQ15M 60155532 IC50 = 19900 nM T60529 CLX65R 60155533 IC50 = 30100 nM T60529 CY1B9U 60155534 IC50 = 9500 nM T60529 CL71GR 60163969 IC50 = 60 nM T60529 CP05UZ 66554464 IC50 = 16100 nM T60529 C97DBL 66695948 IC50 = 1900 nM T60529 C17JAZ 68284084 IC50 = 6400 nM T60529 CH8WL2 70438810 IC50 = 530 nM T60529 CSEA15 70688197 IC50 = 20 nM T60529 C2AX0N 71449035 IC50 = 1000000 nM T60529 CAZ71T 71495779 IC50 > 50000 nM T60529 C5YVD4 71495780 IC50 = 29090 nM T60529 CC0F9V 71495781 IC50 > 50000 nM T60529 C3WYB9 71495782 IC50 = 35360 nM T60529 CO5N4Y 71495783 IC50 > 50000 nM T60529 CK3VM2 71495784 IC50 > 50000 nM T60529 C8JQ0X 71495885 IC50 = 34680 nM T60529 C5L3NI 71495887 IC50 = 38390 nM T60529 CBTR23 71495888 IC50 = 32260 nM T60529 CYEG63 71495889 IC50 > 50000 nM T60529 CQ3T6J 71495988 IC50 = 40390 nM T60529 CXSL48 71495989 IC50 > 50000 nM T60529 C2T8MR 71495990 IC50 > 50000 nM T60529 C90OJI 71495991 IC50 > 50000 nM T60529 CUT0L5 71495992 IC50 = 45880 nM T60529 C82AZY 71495993 IC50 > 50000 nM T60529 C78ZJW 71509612 IC50 > 100000 nM T60529 CXN9L6 71509614 IC50 > 100000 nM T60529 CPN8U4 71550737 IC50 = 2190 nM T60529 C7R5EZ 71571581 IC50 = 7500 nM T60529 C7XMC2 71583324 IC50 = 160 nM T60529 CX18FE 71583325 IC50 = 210 nM T60529 COLY35 71583326 IC50 = 320 nM T60529 CUCE37 71583327 IC50 = 340 nM T60529 C5H2JA 71583438 IC50 = 390 nM T60529 CWRF17 71583439 IC50 = 420 nM T60529 C2OAB4 71583440 IC50 = 170 nM T60529 CCL43F 71583441 IC50 = 240 nM T60529 CB91XC 71583442 IC50 = 390 nM T60529 CK37YJ 71583443 IC50 = 360 nM T60529 C1PH5V 71583444 IC50 = 400 nM T60529 C7T4GM 71583556 IC50 = 440 nM T60529 CK1BH2 71652197 IC50 > 50000 nM T60529 C6IFQ2 71652198 IC50 > 50000 nM T60529 CV6K8P 71652199 IC50 > 50000 nM T60529 CV4NQ3 71652200 IC50 > 50000 nM T60529 CVU9N1 71652201 IC50 > 50000 nM T60529 CA1I3B 71652364 IC50 > 50000 nM T60529 C3XR0J 71652365 IC50 > 50000 nM T60529 CPA68L 71652366 IC50 > 50000 nM T60529 C8E1DW 71652367 IC50 > 50000 nM T60529 CT4RC7 71652368 IC50 = 34980 nM T60529 CVU84Z 71652369 IC50 > 50000 nM T60529 CXVN32 71652528 IC50 > 50000 nM T60529 CY0Q2M 71652529 IC50 > 50000 nM T60529 CTQ6H0 71652530 IC50 > 50000 nM T60529 CT7Z9H 71652531 IC50 = 45060 nM T60529 C5MX2K 71652532 IC50 > 50000 nM T60529 CKY25V 71652533 IC50 = 40560 nM T60529 CYG5R6 71652683 IC50 > 50000 nM T60529 C8RI2F 71652684 IC50 = 39060 nM T60529 C7AYD3 71652685 IC50 > 50000 nM T60529 CEB1P0 71652686 IC50 = 45190 nM T60529 C52OGW 71652687 IC50 > 50000 nM T60529 CPY76V 71682135 IC50 > 100000 nM T60529 CN3O0S 71682136 IC50 = 37000 nM T60529 CQG9Z8 71714062 IC50 = 71400 nM T60529 C2WM6B 71714209 IC50 = 50500 nM T60529 CLS75K 71716000 IC50 > 100000 nM T60529 CYL26P 71718474 IC50 > 100000 nM T60529 CWC7Y9 71720245 IC50 > 100000 nM T60529 CLMV21 73333200 IC50 = 140000 nM T60529 CBTQ18 73333399 IC50 = 300000 nM T60529 CXKH51 73356534 IC50 = 161000 nM T60529 CWY14K 76310400 IC50 = 3610 nM T60529 CL1PM5 76310401 IC50 = 710 nM T60529 CYN6O9 76310402 IC50 = 1350 nM T60529 CZ4J8T 76310403 IC50 = 4210 nM T60529 C9MAL6 76313613 IC50 = 111340 nM T60529 C7B5UG 76314063 IC50 = 18140 nM T60529 C71MXA 76314064 IC50 = 4110 nM T60529 C8PY6T 76317113 IC50 = 389200 nM T60529 CN3IY0 76317622 IC50 = 6650 nM T60529 CW75NC 76317623 IC50 = 19620 nM T60529 C6LPX0 76317624 IC50 = 3280 nM T60529 CR0TN5 76317625 IC50 = 1470 nM T60529 CA7T1F 76317626 IC50 = 1400 nM T60529 CY38AN 76317627 IC50 = 1740 nM T60529 CED02X 76317628 IC50 = 1370 nM T60529 C0YJI7 76317763 IC50 = 580 nM T60529 CWUV56 76320831 IC50 = 188200 nM T60529 CX80WZ 76320832 IC50 = 207360 nM T60529 C8AYK0 76328049 IC50 = 138250 nM T60529 CC7O9K 76328514 IC50 = 2320 nM T60529 C8DQT1 76328515 IC50 = 270 nM T60529 CX9LH5 76328516 IC50 = 2090 nM T60529 C5IME3 76332195 IC50 = 1930 nM T60529 CNPC96 76332196 IC50 = 440 nM T60529 CF17OX 76335317 IC50 = 174720 nM T60529 CL3W1Z 76335832 IC50 = 14930 nM T60529 C7KSB4 78091888 IC50 > 100000 nM T60529 C1GU3V 78091940 IC50 > 100000 nM T60529 CE7N2Q 90643681 IC50 = 24230 nM T60529 C5DLR2 90643682 IC50 = 140450 nM T60529 CO10ZA 90643683 IC50 = 154260 nM T60529 CRFN68 90643684 IC50 = 163240 nM T60529 CQR2T6 90643685 IC50 = 96560 nM T60529 C73HBN 90643686 IC50 = 102660 nM T60529 CS97HW 90643687 IC50 = 89370 nM T60529 CIF45T 90643688 IC50 = 88260 nM T60529 C26ZQJ 90643689 IC50 = 80820 nM T60529 CVTB83 90643690 IC50 = 44350 nM T60529 C9X7IS 90643691 IC50 = 186110 nM T60529 COR58K 90643692 IC50 = 192150 nM T60529 CFO91K 90643693 IC50 = 132320 nM T60529 CLD39A 90643694 IC50 = 38360 nM T60529 CT0BL2 90643695 IC50 = 103520 nM T60529 CDBK93 90643696 IC50 = 115230 nM T60529 CF2KN9 90643697 IC50 = 107250 nM T60529 CX1YR5 90643698 IC50 = 246200 nM T60529 CTF73H 101676817 IC50 = 124400 nM T60529 C9MQW5 118222220 IC50 > 10000 nM T60529 C45NGL 118222276 IC50 > 10000 nM T60529 C91HFT 118222278 IC50 > 30000 nM T60529 C8AMT1 118222288 IC50 > 10000 nM T60529 C7YGX4 118222370 IC50 > 10000 nM T60529 CC3R1W 118705847 IC50 = 17010 nM T60529 CFYD82 118705848 IC50 = 19020 nM T60529 CF7YS2 118705849 IC50 = 41520 nM T60529 CTP28O 118705850 IC50 = 18960 nM T60529 C46XYG 118705851 IC50 = 34530 nM T60529 CP6Q5Z 118705852 IC50 = 10040 nM T60529 C25KZC 118705853 IC50 = 15240 nM T60529 C8ZP5B 118705854 IC50 = 38690 nM T60529 CH8BD1 118705855 IC50 = 64910 nM T60529 C7PU9Q 118706109 IC50 = 57530 nM T60529 CZ6P1A 118706110 IC50 = 40610 nM T60529 CZ41SY 118706111 IC50 = 10760 nM T60529 CAK53T 118706112 IC50 = 17640 nM T60529 CHZQ47 118706113 IC50 = 7230 nM T60529 CO03UN 118706114 IC50 = 105600 nM T60529 CL71XC 118706115 IC50 = 14110 nM T60529 CXZU03 118706116 IC50 = 100300 nM T60529 CI7N0Z 118706117 IC50 = 8750 nM T60529 CA0YD9 118706118 IC50 = 152600 nM T60529 CDPZ58 118706119 IC50 > 500000 nM T60529 CR7PT9 118706120 IC50 = 4630 nM T60529 CFQP30 118706121 IC50 = 3720 nM T60529 C49MZI 118706122 IC50 = 15370 nM T60529 CLE92N 118706123 IC50 = 10360 nM T60529 C23ZNM 118715215 IC50 = 6500 nM T60529 CX9A3J 118715217 IC50 = 117000 nM T60529 CR5WB9 118720945 IC50 > 100000 nM T60529 CL2X8K 118721971 IC50 = 180 nM T60529 CH83RC 118721972 IC50 = 360 nM T60529 CQ7GX9 118721974 IC50 > 4000 nM T60529 CGAI63 118732322 IC50 > 100000 nM T60529 CSH9W4 118732323 IC50 = 99870 nM T60529 CZ1RW7 118732324 IC50 = 91520 nM T60529 CN0YW1 118732325 IC50 = 88380 nM T60529 CO8EN9 118732326 IC50 = 96240 nM T60529 C1BMZ2 118732327 IC50 = 85460 nM T60529 CGT23L 118732328 IC50 > 100000 nM T60529 C3I0PV 118732329 IC50 > 100000 nM T60529 C32HRJ 118732330 IC50 > 100000 nM T60529 C5FNC2 118732331 IC50 > 100000 nM T60529 C8OS5F 118732332 IC50 > 100000 nM T60529 CI4HR8 118732333 IC50 = 100200 nM T60529 C4I6RK 118732334 IC50 > 100000 nM T60529 CVU70J 118732335 IC50 = 86230 nM T60529 CBEH21 118732336 IC50 > 100000 nM T60529 CH7Y4R 118732337 IC50 > 100000 nM T60529 CF1Z6J 118732338 IC50 = 99840 nM T60529 CG01BT 118732339 IC50 = 59360 nM T60529 CH4XL0 118732340 IC50 = 68490 nM T60529 C3WTD0 118732341 IC50 = 78100 nM T60529 C6YXJ5 118732342 IC50 > 100000 nM T60529 C87MQF 118732343 IC50 = 86760 nM T60529 CCEO82 118732344 IC50 > 100000 nM T60529 CW79HI 118732345 IC50 = 90230 nM T60529 C48ZGB 118732346 IC50 > 100000 nM T60529 CC57TX 118732347 IC50 = 96330 nM T60529 CNY30X 118732348 IC50 > 100000 nM T60529 CK3O4I 122182704 IC50 = 40400 nM T60529 CK6AX3 122182705 IC50 = 50600 nM T60529 CKF4H7 122182706 IC50 = 35800 nM T60529 CJ8D7T 122182707 IC50 = 39800 nM T60529 CJ6E4Z 122182708 IC50 = 42800 nM T60529 C5I8SH 122182709 IC50 = 40100 nM T60529 C1VE5G 122182710 IC50 = 54900 nM T60529 C9CE7G 122182711 IC50 = 59900 nM T60529 CW14SV 122182712 IC50 = 50800 nM T60529 CGX21Y 122182713 IC50 = 40800 nM T60529 CI4OQ5 122192740 IC50 = 1800 nM T60529 CP90JH 122192741 IC50 > 100000 nM T60529 CU96HS 122192742 IC50 > 100000 nM T60529 C5Z4RW 122192743 IC50 = 22000 nM T60529 CDN0A3 123278303 IC50 = 8350 nM T60529 CQA34G 127049134 IC50 > 100000 nM T60529 CV64AJ 127049135 IC50 = 89530 nM T60529 CRO71E 127049136 IC50 = 48210 nM T60529 CXMV19 127049150 IC50 = 69250 nM T60529 C8F3NJ 127049474 IC50 = 49760 nM T60529 C3VK2H 127051106 IC50 = 78540 nM T60529 CZ3M1S 127051109 IC50 = 86240 nM T60529 CTW94N 127051121 IC50 > 100000 nM T60529 CT96YA 127051122 IC50 = 96590 nM T60529 C9U5CW 127051123 IC50 > 100000 nM T60529 CAQD52 127051124 IC50 = 74300 nM T60529 CJQM74 127051125 IC50 = 53430 nM T60529 C1NB2H 127051922 IC50 = 39450 nM T60529 C6OBL0 127051923 IC50 > 100000 nM T60529 CB96YL 127051924 IC50 = 84270 nM T60529 C64RNC 127051925 IC50 > 100000 nM T60529 CNH54C 127052535 IC50 = 42160 nM T60529 C62ZJO 127052536 IC50 = 48200 nM T60529 CO4QG9 129886428 IC50 = 10460 nM T60529 C5T4EQ 131801158 IC50 = 104000 nM T60529 C19USV 134134738 IC50 = 206600 nM T60529 CQK60R 134135733 IC50 = 194984.46 nM T60529 C4E7QU 134136565 IC50 = 1548816.62 nM T60529 CX41OZ 134138064 IC50 = 722300 nM T60529 CAEZ47 134138298 IC50 = 229100 nM T60529 C90LTZ 134141655 IC50 = 181970.09 nM T60529 C6U7LZ 134143054 IC50 = 497300 nM T60529 CH86VI 134147676 IC50 = 263026.8 nM T60529 C5XR2B 134152086 IC50 = 380189.4 nM T60529 CJI9Y3 134152691 IC50 = 138038.43 nM T60529 CDV05U 134154144 IC50 = 181970.09 nM T60529 CA08HM 134154737 IC50 = 301995.17 nM T60529 C1GY2T 135156251 EC50 > 10000 nM T60529 CHS9Q1 135401075 IC50 = 1700 nM T60529 CZ0M4A 135407197 IC50 = 4100 nM T60529 C5AXQ9 135411265 IC50 = 430 nM T60529 C5XLH3 135412819 IC50 > 20000 nM T60529 C6Z1ME 135417317 IC50 > 20000 nM T60529 CB2L3G 135419219 IC50 = 1200 nM T60529 CPTI38 135419252 IC50 = 1900 nM T60529 CN3KQ5 135430565 IC50 > 20000 nM T60529 CVR89H 135444615 IC50 = 3100 nM T60529 C1PMI3 135444631 IC50 > 20000 nM T60529 CAH1F2 135461018 IC50 = 12200 nM T60529 C10NPU 135461834 IC50 = 1900 nM T60529 C6P7QT 135464202 IC50 = 9200 nM T60529 CPEX68 135467810 IC50 > 20000 nM T60529 C28NZL 135467819 IC50 = 9900 nM T60529 CJD1E8 135476136 IC50 = 4500 nM T60529 CA8UC6 135476177 IC50 = 14600 nM T60529 C4HW1Z 135480072 IC50 > 20000 nM T60529 CQ29PT 135480085 IC50 > 20000 nM T60529 C8JH3G 135491761 IC50 = 8400 nM T60529 CH9C7U 135493485 IC50 > 20000 nM T60529 CE76OB 135497218 IC50 = 1200 nM T60529 CZOP78 135497261 IC50 > 20000 nM T60529 C9CT1H 135502784 IC50 > 20000 nM T60529 CS9O4H 135502974 IC50 > 200000 nM T60529 CU53ZB 135503592 IC50 = 3200 nM T60529 CK6C8G 135503854 IC50 = 4100 nM T60529 CAB5M3 135503855 IC50 = 13600 nM T60529 CWN8H2 135506078 IC50 > 20000 nM T60529 C5RYH6 135512019 IC50 > 20000 nM T60529 C5Z9ED 135513895 IC50 = 200 nM T60529 CW7YI3 135513937 IC50 = 3600 nM T60529 CL28MS 135515182 IC50 > 20000 nM T60529 C21LGY 135517308 IC50 = 3600 nM T60529 CZ4T5K 135518175 IC50 = 530 nM T60529 CDC4X5 135525549 IC50 = 8400 nM T60529 C2DUW6 135529925 IC50 > 20000 nM T60529 CX9H1L 135532444 IC50 > 100000 nM T60529 CCG7O5 135537152 IC50 > 20000 nM T60529 CH6TK3 135543992 IC50 = 200 nM T60529 CU0OW5 135693491 IC50 = 3640 nM T60529 C2YX9D 135748955 IC50 = 1200 nM T60529 C8K2NT 135786528 IC50 = 5800 nM T60529 CT1C9J 135786531 IC50 = 1200 nM T60529 C3ACW8 135786533 IC50 > 20000 nM T60529 CGBM73 135786534 IC50 = 3600 nM T60529 C1S6KC 135786539 IC50 = 2800 nM T60529 C7OJC8 135786549 IC50 = 3200 nM T60529 C8JCM5 135786553 IC50 = 2800 nM T60529 CX25SL 135786554 IC50 = 300 nM T60529 CHM3Y8 135972420 IC50 = 680 nM T60529 CYSW23 136094858 IC50 > 100000 nM T60529 CFO48N 136094859 IC50 > 100000 nM T60529 CM8Q9X 136152995 IC50 = 155950 nM T60529 CSK95Y 136504263 IC50 = 13 nM T60529 C2IPJ1 137412816 IC50 > 10000 nM T60529 CCYO27 137412823 IC50 > 10000 nM T60529 C52PCB 137412826 IC50 > 10000 nM T60529 C9G2IS 137412832 IC50 > 10000 nM T60529 C9K7QT 137412863 IC50 > 10000 nM T60529 C4LD8H 137632223 IC50 = 70.4 nM T60529 C02ZKT 137632796 IC50 = 43610 nM T60529 C2FA0K 137632978 IC50 = 59230 nM T60529 C0LYA4 137634609 IC50 = 41460 nM T60529 CMH92C 137635036 IC50 > 10000 nM T60529 CC53HT 137637798 IC50 = 47550 nM T60529 C72SBZ 137638298 IC50 = 6750 nM T60529 CJ76FA 137638345 IC50 = 40450 nM T60529 C4WX2T 137638629 IC50 = 113120 nM T60529 CS8KB1 137638984 IC50 = 66.7 nM T60529 C6T1GM 137639040 IC50 > 60000 nM T60529 C8DGE3 137639285 IC50 > 10000 nM T60529 CP1I9Z 137639679 IC50 = 56520 nM T60529 CGQ04J 137641089 IC50 = 74.4 nM T60529 CYV07I 137642019 IC50 = 88.1 nM T60529 CQK8H9 137646026 IC50 = 53080 nM T60529 CZT65P 137647326 IC50 > 60000 nM T60529 C1SOP6 137649486 IC50 > 60000 nM T60529 CJHR31 137649745 IC50 = 43280 nM T60529 CHJ07Q 137649937 IC50 > 10000 nM T60529 COZ38A 137650099 IC50 = 51390 nM T60529 C29KWG 137650898 IC50 = 45350 nM T60529 CILT87 137652137 IC50 = 57260 nM T60529 C3CA7S 137652330 IC50 = 30410 nM T60529 C87VSD 137652535 IC50 = 52670 nM T60529 CE4RY1 137654190 IC50 = 59060 nM T60529 C1ONT8 137659426 IC50 = 36140 nM T60529 C7NE9X 137659718 IC50 > 10000 nM T60529 CPAL37 137661149 IC50 = 95440 nM T60529 C1MKL9 137661257 IC50 = 26250 nM T60529 C80LGK 137661666 IC50 = 134780 nM T60529 CF74TS 137661963 IC50 = 41980 nM T60529 CX06CI 138542656 IC50 > 50000 nM T60529 CX0L1A 139035063 IC50 = 1200 nM T60529 C3ZFV8 145949611 IC50 = 400 nM T60529 CFNO28 145950339 IC50 = 145000 nM T60529 CG37FR 145950583 IC50 = 118000 nM T60529 CCN16Y 145952805 IC50 = 178000 nM T60529 C2FVO7 145953074 IC50 = 152000 nM T60529 CWQ40O 145954141 IC50 = 36110 nM T60529 C19TPY 145958203 IC50 = 201000 nM T60529 CBL1V0 145959229 IC50 = 270 nM T60529 C1BLR8 145959460 IC50 = 137000 nM T60529 C7F1WN 145960726 IC50 = 56000 nM T60529 C6R3AF 145960841 IC50 = 56000 nM T60529 CRV1U7 145962585 IC50 = 56000 nM T60529 CBG7X0 145963101 IC50 = 56000 nM T60529 C65QKS 145963415 IC50 = 56000 nM T60529 CUXQ13 145971245 IC50 = 167000 nM T60529 C8U9TX 145971276 IC50 = 120000 nM T60529 CZPC04 145982667 IC50 = 32160 nM T60529 C0LU3T 145982976 IC50 = 39450 nM T60529 C20AWS 145983008 IC50 = 27890 nM T60529 CA8U6O 145983125 IC50 = 43200 nM T60529 CGZ73L 145983279 IC50 > 50000 nM T60529 CR61XP 145983281 IC50 = 49640 nM T60529 CP54SE 145983381 IC50 = 47480 nM T60529 C0HE8J 145983476 IC50 = 25520 nM T60529 C2W1PX 145983528 IC50 = 44820 nM T60529 CMTE25 145983596 IC50 = 41080 nM T60529 C0LF5R 145983962 IC50 = 42050 nM T60529 CAB1M0 145984018 IC50 = 46450 nM T60529 CDW7Q2 145984214 IC50 > 50000 nM T60529 C09ZYR 145984318 IC50 = 32930 nM T60529 C6RS2D 145984423 IC50 = 43200 nM T60529 CUY3T9 145984477 IC50 = 32930 nM T60529 CB9X6S 145984519 IC50 = 33760 nM T60529 C8-MAR-07 145984539 IC50 = 44800 nM T60529 CXPK46 145984992 IC50 > 50000 nM T60529 C3KEW1 145985004 IC50 = 39120 nM T60529 C50TGP 145985054 IC50 > 50000 nM T60529 C1LEX8 145985067 IC50 = 40930 nM T60529 CTE68V 145985355 IC50 = 33120 nM T60529 CRIT31 145985451 IC50 = 41340 nM T60529 CL6ZW3 145985573 IC50 = 36850 nM T60529 C7FWH1 145985695 IC50 = 45040 nM T60529 C1T2XR 145985744 IC50 = 41240 nM T60529 C2RO7H 145986163 IC50 = 30160 nM T60529 CBEG25 145986220 IC50 = 27620 nM T60529 CV6BD5 145986241 IC50 = 29740 nM T60529 CU5E9G 155511187 IC50 = 450 nM T60529 CCIZ41 155512205 IC50 = 506.8 nM T60529 C3JX1B 155512689 IC50 = 7770 nM T60529 C3R8LP 155512734 IC50 = 73.27 nM T60529 CM0OK6 155514659 IC50 = 2890 nM T60529 CZB64G 155514739 IC50 = 7750 nM T60529 CAZ16P 155514890 IC50 = 29350 nM T60529 CK21YX 155515749 IC50 = 370 nM T60529 CM0O8D 155516306 IC50 = 310 nM T60529 CFD4A0 155516566 IC50 = 5590 nM T60529 C5VNH3 155516647 IC50 = 15460 nM T60529 CY3DR9 155516693 IC50 = 876 nM T60529 C3P4MO 155517441 IC50 = 540 nM T60529 CQK2J3 155518007 IC50 = 32060 nM T60529 CCH5E8 155519683 IC50 = 2720 nM T60529 C02HAV 155521349 IC50 = 13010 nM T60529 C3YGK8 155521606 IC50 > 30000 nM T60529 CQ3N6D 155521710 IC50 = 204.72 nM T60529 CPKS90 155521809 IC50 = 16500 nM T60529 C98MBO 155522237 IC50 = 9570 nM T60529 C69GCU 155522308 IC50 > 100000 nM T60529 CB41LZ 155522446 IC50 = 28520 nM T60529 CSY34V 155523202 IC50 = 161.06 nM T60529 C4PGA5 155523362 IC50 > 100000 nM T60529 CA8Q1L 155523402 IC50 = 7200 nM T60529 CF82YG 155523642 IC50 = 13160 nM T60529 C69ECX 155524453 IC50 = 180700 nM T60529 C30OZI 155527652 IC50 = 14150 nM T60529 CK7EU9 155527685 IC50 = 166300 nM T60529 C95UOG 155528389 IC50 = 30000 nM T60529 C80BRK 155528880 IC50 = 30790 nM T60529 CB9M1X 155529539 IC50 = 6070 nM T60529 C2GLH7 155529640 IC50 = 5200 nM T60529 CB4WF1 155530728 IC50 = 700 nM T60529 C1QXU2 155530946 IC50 = 878.8 nM T60529 CIJ3G0 155531569 IC50 = 15000 nM T60529 C51EJF 155531595 IC50 > 100000 nM T60529 CUL96H 155531758 IC50 = 460 nM T60529 CRD14L 155532032 IC50 = 169.28 nM T60529 CD94TA 155534770 IC50 = 13200 nM T60529 C6RB5J 155534811 IC50 = 43720 nM T60529 CA69IG 155534995 IC50 = 15620 nM T60529 CE3VB4 155535321 IC50 = 103000 nM T60529 C2PN5F 155536316 IC50 = 104400 nM T60529 C2Z7GX 155537370 IC50 = 141800 nM T60529 CNU2C0 155544451 IC50 > 100000 nM T60529 CEZ3U5 155544780 IC50 = 115.64 nM T60529 C53BXM 155545107 IC50 = 104300 nM T60529 CK3EW2 155545512 IC50 > 100000 nM T60529 CB9V4N 155545715 IC50 = 270 nM T60529 C30NDT 155546179 IC50 = 104.17 nM T60529 C02VES 155546488 IC50 > 100000 nM T60529 CVP4G7 155547475 IC50 = 64.74 nM T60529 C4CY2L 155548534 IC50 = 132100 nM T60529 C7IES3 155548701 IC50 = 155300 nM T60529 CYDP17 155551847 IC50 = 676.9 nM T60529 CZO59G 155552038 IC50 = 99600 nM T60529 CG1U2I 155553094 IC50 = 600 nM T60529 CYG31B 155553429 IC50 = 210 nM T60529 C3CG7H 155553481 IC50 = 27220 nM T60529 C7BM0W 155553539 IC50 = 9680 nM T60529 CB18OG 155554424 IC50 = 71970 nM T60529 CHGI70 155557383 IC50 = 94300 nM T60529 CCV8M6 155558071 IC50 = 103800 nM T60529 CERZ85 155558072 IC50 = 4020 nM T60529 C4V6GB 155558213 IC50 > 100000 nM T60529 CHI7P2 155558802 IC50 = 7080 nM T60529 CVGD95 155559759 IC50 = 123.15 nM T60529 CF4W8Y 155559976 IC50 = 390 nM T60529 CK9PR5 155560364 IC50 = 9040 nM T60529 C50XAB 155562173 IC50 = 6220 nM T60529 C13BZU 155563007 IC50 = 8890 nM T60529 CP8BG6 155563791 IC50 = 7920 nM T60529 CX12MT 155563845 IC50 = 240 nM T60529 C53AWR 155563991 IC50 = 162.97 nM T60529 CV4I2Q 155564403 IC50 = 27690 nM T60529 CF7G4U 155565228 IC50 = 65390 nM T60529 C79ZDF 155566047 IC50 = 8630 nM T60529 C28TBL 155567336 IC50 = 513 nM T60529 CU3F4D 155568632 IC50 = 6410 nM T60529 C70ZUA 155569262 IC50 > 100000 nM T60529 CC35YL 11335338 IC50 > 100000 nM T60529 CL4VS1 118222242 IC50 > 100000 nM T60529 CQF61C 118720946 IC50 > 100000 nM T60529 D00AII 5281727 IC50 = 700 nM T60529 D00YGP 11536337 IC50 = 30100 nM T60529 D01MFK 9906892 IC50 = 14000 nM T60529 D01SNR 208910 IC50 = 25000 nM T60529 D01WLL 11460185 IC50 = 3620 nM T60529 D02FEF 404378 IC50 = 383360 nM T60529 D02FGY 44434501 IC50 = 10600 nM T60529 D03FXI 564225 IC50 = 141250 nM T60529 D03LOG 5280450 IC50 = 13000 nM T60529 D03NMM 46843035 IC50 > 100000 nM T60529 D03VUQ 404202 IC50 = 148200 nM T60529 D04HRS 404195 IC50 > 100000 nM T60529 D04YPP 9991673 IC50 = 90 nM T60529 D05IWY 5464078 IC50 = 800 nM T60529 D05JRZ 67316 IC50 = 31570 nM T60529 D06DRL 44475843 IC50 = 2260 nM T60529 D06GUJ 44428631 IC50 = 600 nM T60529 D06WML 10377376 IC50 = 50 nM T60529 D06YGF 5281787 IC50 = 58000 nM T60529 D06ZRX 5281717 IC50 = 1400 nM T60529 D07JDC 10364 IC50 = 4000 nM T60529 D07LUJ 64945 IC50 = 210000 nM T60529 D07QIU 625902 IC50 = 313830 nM T60529 D07STC 44434500 IC50 = 19800 nM T60529 D08UOX 5281148 IC50 = 66000 nM T60529 D09DMR 44456679 IC50 = 63590 nM T60529 D0BO9W 11150126 IC50 = 5340 nM T60529 D0C5SV 5280934 Ki = 4000 nM T60529 D0EI8V 45268661 IC50 = 62000 nM T60529 D0F3UR 690836 IC50 = 190470 nM T60529 D0F6CD 5202 IC50 > 400000 nM T60529 D0FQ3N 5748382 IC50 > 100000 nM T60529 D0G3TK 5280863 IC50 > 100000 nM T60529 D0J1AW 405560 IC50 = 38200 nM T60529 D0JT8Y 21177358 IC50 = 105630 nM T60529 D0L6TP 11277773 IC50 = 18360 nM T60529 D0LJ7R 15345559 IC50 = 9700 nM T60529 D0M5MI 4306515 IC50 = 8.9 nM T60529 D0O7SM 5281514 IC50 = 14000 nM T60529 D0QV6M 4292 IC50 > 66000 nM T60529 D0S2II 308405 IC50 = 108340 nM T60529 D0S7LD 5326145 IC50 > 100000 nM T60529 D0SJ2Q 10494 IC50 = 380000 nM T60529 D0T2SD 21862824 IC50 = 63220 nM T60529 D0T4VL 9908776 IC50 > 1000000 nM T60529 D0T9QW 33675 IC50 = 2800 nM T60529 D0UH3D 49837499 IC50 = 24000 nM T60529 D0V3PG 128861 IC50 = 90000000 nM T60529 D0V7AA 9064 IC50 = 36700 nM T60529 D0V9EN 689043 IC50 > 400000 nM T60529 D0VF6F 10244543 IC50 = 410 nM T60529 D0X6RO 404324 IC50 = 159070 nM T60529 D0Y1YR 442793 IC50 = 129000 nM T60529 D0Y9ZO 21862753 IC50 = 80200 nM T60529 D0YZ5G 5281416 IC50 = 57000 nM T60529 D0Z1WF 405489 IC50 > 100000 nM T63024 D0G5UB 2161 IC50 = 851.14 nM T63024 D0OB0F 5328940 IC50 = 471 nM T63024 D02XNW 5494449 IC50 = 6.22 nM T63024 D09JEJ 24748573 IC50 = 35 nM T63024 D0E3TC 44259 IC50 = 2.18 nM T63024 D03BNU 59604787 IC50 > 10000 nM T63024 D09FGW 56646218 IC50 = 1 nM T63024 D0T3ME 156422 IC50 > 30000 nM T63024 CJ2T3N 10023121 IC50 = 383 nM T63024 C0IVL9 10347359 IC50 = 6 nM T63024 CW5C9X 11186250 IC50 > 3162.28 nM T63024 CM21YJ 11453049 IC50 > 3162.28 nM T63024 CACS26 11561968 Ki > 2000 nM T63024 CGX96V 11626927 IC50 = 72 nM T63024 CJ9KN7 11683817 IC50 > 10000 nM T63024 CU0E8O 11690457 Ki > 2000 nM T63024 CB0AP2 11705863 Ki > 10000 nM T63024 CM7S0Z 12852146 IC50 = 400 nM T63024 C41KUL 15571856 IC50 = 524.81 nM T63024 C5VPH9 16129448 IC50 = 1070 nM T63024 C7YG1N 24759534 IC50 < 10 nM T63024 CLBP72 24798571 IC50 > 4000 nM T63024 CU19EF 44231127 IC50 = 8 nM T63024 CI3BA2 44462961 IC50 = 820 nM T63024 C3XY7U 44464266 IC50 = 11 nM T63024 CQ8BA1 44464268 IC50 = 3 nM T63024 CLI16E 44465026 IC50 = 8 nM T63024 C6RXW1 44465027 IC50 = 9 nM T63024 C8CF6N 44465029 IC50 = 3200 nM T63024 CEK2D3 44465285 IC50 = 4 nM T63024 C6M9IQ 44465820 IC50 = 2 nM T63024 CJW93H 44466599 IC50 = 28 nM T63024 C3VRO9 44557921 IC50 > 10000 nM T63024 CEQN27 52936621 Ki > 1000 nM T63024 C8NA4L 53384644 IC50 > 30000 nM T63024 C03XBT 57328467 EC50 = 139 nM T63024 CXJ35L 57328543 EC50 = 35 nM T63024 CCF61V 57328544 EC50 = 34 nM T63024 C39KXI 57328545 EC50 = 17 nM T63024 C2TC6M 59225246 IC50 = 63 nM T63024 C8K5QN 59225250 IC50 = 6 nM T63024 CT70FI 59225251 IC50 = 2 nM T63024 COCB23 59225272 IC50 = 7 nM T63024 CAK48J 59225283 IC50 = 16 nM T63024 CH0G1X 59225285 IC50 = 15 nM T63024 C1W9GK 59225297 IC50 = 3 nM T63024 C3SBA4 59225303 IC50 = 8 nM T63024 C8TQB4 59225307 IC50 > 1000 nM T63024 CT5OV9 59225334 IC50 = 13 nM T63024 CHV18S 59225349 IC50 = 9 nM T63024 C7FQD2 59225366 IC50 = 110 nM T63024 CM48WR 59225375 IC50 = 2 nM T63024 CXJC43 59225411 IC50 = 2 nM T63024 C4K7PD 59225430 IC50 > 1000 nM T63024 CXJ63M 59603829 IC50 < 10 nM T63024 CQEU96 59603842 IC50 < 1 nM T63024 COH62U 60097413 IC50 > 10000 nM T63024 C1MR8Q 60097495 IC50 > 1000 nM T63024 C37NKO 67129970 IC50 > 10000 nM T63024 CK80LJ 67130050 IC50 > 10000 nM T63024 CV63UL 67240318 IC50 > 10000 nM T63024 C7GRV2 68755406 IC50 > 10000 nM T63024 C5DGR9 69036886 IC50 = 10000 nM T63024 C6F4QX 70681026 IC50 = 151 nM T63024 CQ63HX 70681027 IC50 = 231 nM T63024 CR2QO7 70681028 IC50 = 106 nM T63024 CRZ36H 70681029 IC50 = 12000 nM T63024 CZ4OY5 70681030 IC50 = 8 nM T63024 CU6NE9 70681031 IC50 = 59 nM T63024 CPOV92 70681032 IC50 = 3 nM T63024 COHI26 70681033 EC50 = 12 nM T63024 C48POI 70683150 IC50 = 468 nM T63024 C25FGR 70683151 IC50 = 345 nM T63024 CSN7L4 70683152 IC50 = 178 nM T63024 C6XO5Q 70683153 IC50 = 288 nM T63024 CW8LF0 70683154 IC50 = 1520 nM T63024 C7EH1D 70683155 EC50 = 11 nM T63024 C5I7DW 70685226 IC50 = 426 nM T63024 COYD53 70685227 IC50 = 2740 nM T63024 CU47OG 70685228 IC50 = 257 nM T63024 CZ6NH0 70685229 IC50 = 388 nM T63024 CE65KV 70685230 IC50 = 213 nM T63024 CRK92N 70685231 EC50 = 14 nM T63024 CA57VF 70685232 EC50 = 26 nM T63024 CID9O3 70685233 IC50 = 4 nM T63024 CN2O6T 70687384 IC50 = 229 nM T63024 C4Q5MO 70687385 IC50 = 196 nM T63024 CA0FE8 70687386 EC50 = 111 nM T63024 CQH9A0 70687387 EC50 = 73 nM T63024 CMA7J1 70687388 EC50 = 6 nM T63024 CWD19I 70689442 IC50 = 2290 nM T63024 CW9O7S 70689443 IC50 = 105 nM T63024 CS7LM1 70689444 IC50 = 65 nM T63024 C1MSF8 70689445 IC50 = 233 nM T63024 CD5V2S 70689446 IC50 = 162 nM T63024 CEGM27 70689447 EC50 = 20 nM T63024 C80CWD 70689448 EC50 = 8 nM T63024 CQ1X4K 70691555 IC50 = 335 nM T63024 CN15SY 70691556 IC50 = 4 nM T63024 CO9KZ3 70693645 IC50 = 9550 nM T63024 CG9PD4 70695751 IC50 = 1220 nM T63024 C0B7XU 70695752 IC50 = 10300 nM T63024 CC6ZN8 70695753 IC50 = 1410 nM T63024 CP3G9T 70695755 IC50 = 111 nM T63024 CH2YA1 70695756 IC50 = 93 nM T63024 C47HZW 70695757 IC50 = 192 nM T63024 CL71AV 70695758 IC50 = 39 nM T63024 C2EI9Z 70695759 EC50 = 25 nM T63024 CZ4W6K 70695760 EC50 = 84 nM T63024 CS37NT 71450663 IC50 = 22 nM T63024 CF4P1N 71450664 IC50 > 10000 nM T63024 C2NCX1 71450665 IC50 = 7 nM T63024 CB9H5Y 71450666 IC50 = 7 nM T63024 CO7M9X 71452497 IC50 > 1000 nM T63024 C9I5GF 71454257 IC50 = 3600 nM T63024 C8OWL6 71456015 IC50 = 8 nM T63024 C4QUL2 71456016 IC50 = 450 nM T63024 C6E7MH 71457819 IC50 = 4300 nM T63024 CID65O 71459725 IC50 = 430 nM T63024 CYL46C 71459726 IC50 = 7 nM T63024 CD1W8C 71459727 IC50 = 4 nM T63024 CH83WB 71461445 IC50 = 10 nM T63024 CYN6R5 71461446 IC50 = 9 nM T63024 CET01R 71463176 IC50 = 560 nM T63024 CE9UA2 71463177 IC50 > 10000 nM T63024 C75RVU 71463178 IC50 = 60 nM T63024 C0DL3F 72698602 IC50 < 1 nM T63024 C42MXW 76310923 IC50 = 46 nM T63024 C0MR6F 76310924 IC50 = 136 nM T63024 CJ3I5E 76310925 IC50 = 1040 nM T63024 C6EI1G 76310926 IC50 = 256 nM T63024 CVP8Z4 76310927 IC50 = 129 nM T63024 C9MG7U 76314564 IC50 = 78 nM T63024 CU8EW0 76318141 IC50 = 759 nM T63024 C80VJZ 76318142 IC50 = 98 nM T63024 C6ZOM5 76321826 IC50 = 37 nM T63024 C5MRE6 76321827 IC50 = 268 nM T63024 CZ0XB7 76321828 IC50 = 1050 nM T63024 C1BJ5I 76321829 IC50 > 30000 nM T63024 C8Z6XR 76325460 IC50 = 2170 nM T63024 CKZ4F9 76325461 IC50 = 460 nM T63024 CTA86L 76325462 IC50 = 89 nM T63024 C9B2NA 76325463 IC50 = 859 nM T63024 CLF2S7 76325464 IC50 = 1800 nM T63024 CI7WT3 76325465 IC50 = 49 nM T63024 CT1R6E 76329005 IC50 = 7 nM T63024 CT4FE5 76329006 IC50 = 650 nM T63024 C8ZTP6 76332688 IC50 = 203 nM T63024 C0PRE8 76336290 IC50 = 128 nM T63024 CF1JW0 76336291 IC50 = 30 nM T63024 C1HW4B 89735655 IC50 < 10 nM T63024 CC23OD 91970516 IC50 = 0.06 nM T63024 CQCX41 118737057 IC50 > 10000 nM T63024 CTW92Q 121230617 IC50 = 13 nM T63024 CZ71IR 124108661 IC50 = 1.3 nM T63024 CWS5C4 129245211 IC50 = 372 nM T63024 CH91ON 129245363 IC50 = 9 nM T63024 C6A1LP 129245450 IC50 = 273 nM T63024 COKE50 129245476 IC50 = 764 nM T63024 CA2N5C 129245517 IC50 = 50 nM T63024 C0E2RU 129245526 IC50 = 2270 nM T63024 C9J8HZ 129245530 IC50 = 148 nM T63024 C52PNC 129245623 IC50 = 391 nM T63024 CL21HY 129245681 IC50 = 115 nM T63024 C1QKC7 129245769 IC50 = 34 nM T63024 CEYK58 129245795 IC50 = 5 nM T63024 CFP0G6 129245828 IC50 = 2490 nM T63024 COR37Y 129245842 IC50 = 72 nM T63024 CKB5C8 129245918 IC50 = 58 nM T63024 CQJK71 129246093 IC50 = 2 nM T63024 C0GC7N 129246130 IC50 = 55 nM T63024 C09MDW 129260549 IC50 = 2660 nM T63024 CCF8W2 129261617 IC50 = 10 nM T63024 CG5O2J 129261641 IC50 = 15 nM T63024 CPEA28 130275058 IC50 = 2300 nM T63024 C1BPS0 130275075 IC50 = 290 nM T63024 CSQ0O5 130275093 IC50 = 760 nM T63024 CS8YR1 130275108 IC50 = 550 nM T63024 CCWF83 130275116 IC50 = 300 nM T63024 CJ4GK2 130275332 IC50 = 630957.34 nM T63024 CYHA01 130275488 IC50 = 2290.87 nM T63024 CAT2Q7 130275498 IC50 = 1700 nM T63024 C7S0KD 130275500 IC50 = 1800 nM T63024 CU8IR7 130275554 IC50 = 4600 nM T63024 C6GSW1 130276189 IC50 = 570 nM T63024 C6HY7G 130276200 IC50 = 524807.46 nM T63024 C9G2SC 130276225 IC50 = 750 nM T63024 C7NCV5 130276229 IC50 = 270 nM T63024 CZ9K7R 130276230 IC50 = 830 nM T63024 CD6QO8 130276741 IC50 = 860 nM T63024 CR43KG 130276782 IC50 = 830 nM T63024 CS16TD 130276801 IC50 = 398.11 nM T63024 C1NWB5 130276805 IC50 = 490 nM T63024 CJ2T7Z 130276806 IC50 = 1900 nM T63024 CAQ89B 130276808 IC50 = 750 nM T63024 C90IYP 130276898 IC50 = 12000 nM T63024 COA70I 130276966 IC50 = 790 nM T63024 CPAX52 130276970 IC50 = 440 nM T63024 C8M6VS 130289650 IC50 = 537.03 nM T63024 C1NL4U 130290291 IC50 = 1900 nM T63024 CM65GQ 130290300 IC50 = 1300 nM T63024 CV0TH9 132000066 EC50 = 53900 nM T63024 C5UOY0 136266076 IC50 = 201 nM T63024 C8KJ9Z 137479135 IC50 = 1140 nM T63024 CVHF30 137479140 IC50 = 388 nM T63024 C7B4NR 137479154 IC50 = 5070 nM T63024 CO3NT9 137553174 IC50 = 1000 nM T63024 CI1E8V 137634241 IC50 = 7610 nM T63024 CM07EU 145714274 IC50 = 1 nM T63024 C9ISH6 145925685 IC50 = 30 nM T63024 C1A3HL 145988072 IC50 = 489.78 nM T63024 CT4M9E 145989247 IC50 = 1096.48 nM T63024 C7CH9V 146014951 IC50 = 2 nM T63024 CJB1R5 155511461 IC50 = 2 nM T63024 CV36FS 155512885 IC50 = 188 nM T63024 C2MD1Q 155513187 IC50 > 10000 nM T63024 C80CTM 155520004 IC50 = 1210 nM T63024 CZ0WO7 155523990 IC50 = 2 nM T63024 CHMV49 155525041 IC50 = 93 nM T63024 C82MLZ 155526827 IC50 = 29 nM T63024 CK2RM8 155528214 IC50 = 16700 nM T63024 CH0S4T 155530766 IC50 < 100 nM T63024 C8O6WA 155542495 IC50 = 1060 nM T63024 CHD09S 155543566 IC50 = 7 nM T63024 C2Y4AG 155546383 IC50 = 5 nM T63024 C6JWS0 155560801 IC50 = 281 nM T63024 CQRO74 155567366 IC50 = 98 nM T63024 D00ERW 44444843 Ki > 1525 nM T63024 D03BJF 44465558 IC50 = 6 nM T63024 D06ZIO 44464263 IC50 = 19 nM T63024 D0J3LR 11634725 Ki > 10000 nM T63024 D0RG0Z 10077147 IC50 = 6 nM T22496 CT6M5I 210546 IC50 > 10000 nM T22496 CXC6Y0 720645 EC50 = 50000 nM T22496 C9GY3O 720655 IC50 = 1310 nM T22496 C96IYT 720660 IC50 = 2210 nM T22496 CSO6D3 1092394 IC50 = 1200 nM T22496 C3Y8MD 1560402 EC50 = 50000 nM T22496 CQJ8Z2 1569268 EC50 = 50000 nM T22496 C73NFT 7137844 IC50 = 2740 nM T22496 C1JN0B 21029584 IC50 > 10000 nM T22496 CTB2X0 23631966 IC50 = 1070 nM T22496 CH9O0I 23631971 IC50 = 3440 nM T22496 C2PE8I 23631972 IC50 = 710 nM T22496 CW70BU 23632009 IC50 = 4480 nM T22496 C4WKE6 23827771 IC50 > 10000 nM T22496 CGJ79Y 24742049 IC50 > 10000 nM T22496 CNW76J 24742050 IC50 = 3630 nM T22496 C7EK9G 24742051 IC50 = 10500 nM T22496 CY7M9A 24742052 IC50 > 10000 nM T22496 CV3PW8 24742053 IC50 > 10000 nM T22496 C50CBM 24742055 IC50 = 5260 nM T22496 CI6E0R 24742056 IC50 = 6380 nM T22496 CA5TR4 24742057 IC50 > 15800 nM T22496 CRJ6C2 24742059 IC50 = 1110 nM T92834 CWV9Q2 10477531 IC50 = 1470 nM T92834 CHG02V 10478612 IC50 = 950 nM T92834 C0R5QL 10894433 IC50 = 350 nM T92834 C57OXT 11102540 IC50 = 970 nM T92834 CA43HK 11732287 IC50 = 470 nM T94823 D0Y7ZD 137 Ki = 960000 nM T94823 D01XGX 178060 IC50 > 100000 nM T94823 C82BHU 447280 IC50 = 4900 nM T94823 C8EK7G 9835053 IC50 > 10000 nM T94823 C0Q7BK 10127057 IC50 > 10000 nM T94823 C4U3IC 10144962 IC50 > 10000 nM T94823 C5P0AO 10238227 IC50 > 10000 nM T94823 C3FB4T 10310021 IC50 > 10000 nM T94823 C1YO9B 10375752 Ki = 270 nM T94823 C4OC6P 10455620 IC50 > 10000 nM T94823 C1WKE4 10455621 IC50 > 10000 nM T94823 CH1DG5 10478099 IC50 > 10000 nM T94823 CB3I6Y 10521264 IC50 > 2000000 nM T94823 CN9M6R 10592387 IC50 = 59000 nM T94823 C8PC9N 10624384 IC50 = 110000 nM T94823 CTSJ57 10665335 IC50 > 2000000 nM T94823 CAH46W 10672283 IC50 = 29000 nM T94823 C0YD1X 10687736 IC50 = 410000 nM T94823 C7JWD3 11476287 IC50 > 10000 nM T94823 CMYN65 11526865 IC50 > 40000 nM T94823 CZ35WN 11533932 IC50 > 40000 nM T94823 CPR71X 11540951 IC50 > 40000 nM T94823 C98GDW 11541277 IC50 > 40000 nM T94823 CBR9K8 11541314 IC50 > 40000 nM T94823 CY0A7J 11570138 IC50 > 40000 nM T94823 CQU80H 11576569 IC50 > 40000 nM T94823 CW94NS 11577331 IC50 > 40000 nM T94823 CQ86GI 11577431 IC50 > 40000 nM T94823 CAZL49 11584650 IC50 > 40000 nM T94823 C5JYV7 11591936 IC50 > 40000 nM T94823 CQL5S8 11613750 IC50 > 40000 nM T94823 C7YKC0 11628195 IC50 > 40000 nM T94823 CXG1B4 11649741 IC50 > 40000 nM T94823 C3Y7EL 11678025 IC50 > 40000 nM T94823 CIEJ54 11720809 IC50 > 40000 nM T94823 CN96PD 11724034 IC50 = 2200 nM T94823 C2WUP4 11794649 IC50 = 2200 nM T94823 C0H8OB 24776705 IC50 > 10000 nM T94823 C24GLZ 24776939 IC50 > 10000 nM T94823 C6LD2J 24777439 IC50 > 10000 nM T94823 CK8EL5 24777568 IC50 > 10000 nM T94823 CQ20PV 24777692 IC50 > 10000 nM T94823 C1WF3I 24777804 IC50 > 10000 nM T94823 C3IS2X 44316877 IC50 = 1700000 nM T94823 C6ITG5 44316896 IC50 > 2000000 nM T94823 CS02PC 44317216 IC50 = 130000 nM T94823 CSN27E 44445042 IC50 > 10000 nM T94823 CGN61Q 44445047 IC50 > 10000 nM T94823 CYW8E3 44445051 IC50 > 10000 nM T94823 CRG64M 44445053 IC50 > 10000 nM T94823 C6ZID3 44445055 IC50 > 10000 nM T94823 C72KOR 44445057 IC50 > 10000 nM T94823 C0RTA6 44445060 IC50 > 10000 nM T94823 CIK8G3 44445063 IC50 > 10000 nM T94823 CN05VX 44445065 IC50 > 10000 nM T94823 COA90R 44445067 IC50 > 10000 nM T94823 CX5M9O 49796392 Ki = 1100000 nM T94823 CZ7A9E 49796933 IC50 > 100000 nM T94823 CBD8K2 49796942 IC50 > 100000 nM T94823 CI25XP 49796945 IC50 > 100000 nM T94823 C8WYA5 49796953 IC50 > 100000 nM T94823 CQH86V 49796955 IC50 > 100000 nM T94823 C5W6LY 70681316 IC50 > 10000 nM T94823 CVYH31 70689717 IC50 > 10000 nM T94823 D0CG7Q 10336627 IC50 = 660 nM T94823 D0T3AE 1005 Ki = 8.5 nM T18664 D0X5SD 3117 IC50 = 1258.93 nM T18664 D0CW8S 71657619 IC50 = 2.2 nM T18664 D0JQ9Z 575125 IC50 = 912.01 nM T18664 C3KU4J 7347 IC50 = 12302.69 nM T18664 CC4TF8 7648 IC50 = 11220.18 nM T18664 CB4L9P 12704 IC50 > 1000000 nM T18664 CMC1D0 12892 IC50 = 218.78 nM T18664 CK01EP 13436 IC50 = 1600 nM T18664 CWPE53 13662 IC50 = 15900 nM T18664 CXD5C3 14550 IC50 = 4170 nM T18664 C3KEJ7 15399 IC50 = 14100 nM T18664 C4WGQ6 15400 IC50 = 7240 nM T18664 CT7B0H 16244 IC50 > 1000000 nM T18664 CRXE23 16245 IC50 = 60255.96 nM T18664 CPVM03 18156 IC50 = 2030 nM T18664 CJ6R0G 19989 IC50 = 2690 nM T18664 CXV2S5 20992 IC50 = 1700 nM T18664 CYG8I5 25057 IC50 = 9549.93 nM T18664 CI1N8E 30054 IC50 = 109.65 nM T18664 CUAH61 70261 IC50 = 24500 nM T18664 CFZ4W0 70362 IC50 > 1000000 nM T18664 C81NEO 74204 IC50 = 5140 nM T18664 C3WP1X 81734 IC50 = 12900 nM T18664 CW83UB 82747 IC50 = 741.31 nM T18664 CBCW47 96153 IC50 = 5180 nM T18664 CQV87B 96758 IC50 = 4340 nM T18664 CV4CP1 97695 IC50 = 6920 nM T18664 CNXC25 101342 IC50 = 2390 nM T18664 CD60TZ 123301 IC50 = 4370 nM T18664 CS4N9G 126214 IC50 = 2240 nM T18664 CM9P7S 139950 IC50 = 7943.28 nM T18664 C4IRY2 164676 IC50 = 48000 nM T18664 C12API 224621 IC50 = 5754.4 nM T18664 CD8O5B 225451 IC50 > 1000000 nM T18664 C84BNY 225452 IC50 > 1000000 nM T18664 C2KSN1 229985 IC50 = 14791.08 nM T18664 CI93OA 235603 IC50 = 2630.27 nM T18664 C3LM0H 236788 IC50 = 5750 nM T18664 CSN4G0 239576 IC50 = 28800 nM T18664 C69ONP 243296 IC50 = 7610 nM T18664 CP9C8D 247652 IC50 = 2750 nM T18664 CN7BU2 248003 IC50 = 2820 nM T18664 C6N1RA 270740 IC50 = 19952.62 nM T18664 C4M0BH 285275 IC50 > 1000000 nM T18664 C8OKS7 289457 IC50 = 204173.79 nM T18664 CB73CH 305201 IC50 = 2880 nM T18664 CD1W3N 308434 IC50 = 6600 nM T18664 CE2PB0 329124 IC50 = 2398.83 nM T18664 C43HCK 349626 IC50 = 23988.33 nM T18664 CPM6S8 355227 IC50 = 9549.93 nM T18664 C16VBD 512831 IC50 = 3550 nM T18664 C2ZO3H 522624 IC50 = 2820 nM T18664 CQ76DG 555841 IC50 = 9700 nM T18664 CIK0F2 599019 IC50 = 5010 nM T18664 CUB84X 606562 IC50 = 20892.96 nM T18664 C3EZ5G 619828 IC50 = 9549.93 nM T18664 C8O7SW 684261 IC50 = 77624.71 nM T18664 CB5YI4 691987 IC50 > 1000000 nM T18664 C2T3HR 704937 IC50 = 2000 nM T18664 CM87FU 708576 IC50 > 1000000 nM T18664 CZP2I7 708855 IC50 = 4270 nM T18664 CPD14Q 709265 IC50 = 2920 nM T18664 CH0F9V 766352 IC50 > 1000000 nM T18664 C8GB4W 782503 IC50 > 1000000 nM T18664 CZ4SQ3 782978 IC50 > 1000000 nM T18664 CP04GF 783204 IC50 > 1000000 nM T18664 CYXZ62 812266 IC50 = 31622.78 nM T18664 CTHK18 895402 IC50 > 1000000 nM T18664 CY82IZ 930984 IC50 = 2340 nM T18664 CH5US0 974575 IC50 = 30902.95 nM T18664 C8QFC3 1075551 IC50 > 500000 nM T18664 CW3M4V 1109251 IC50 > 1000000 nM T18664 CUXF32 1130422 IC50 > 500000 nM T18664 C85VNI 1171867 IC50 > 500000 nM T18664 C85WRE 1373945 IC50 > 500000 nM T18664 C6MV7A 1373946 IC50 > 500000 nM T18664 C5T7RG 1438040 Ki = 8600 nM T18664 COR8N4 1446077 IC50 = 24300 nM T18664 CHNJ13 1532212 IC50 = 100000 nM T18664 C3ASC0 2019899 IC50 = 965 nM T18664 C0KTS1 2189777 IC50 > 1000000 nM T18664 C59GIY 2193280 IC50 = 19498.45 nM T18664 CIUM60 2732146 IC50 = 5890 nM T18664 CA59XF 2896608 IC50 = 29512.09 nM T18664 C9I3ZQ 3017401 IC50 = 24000 nM T18664 CM21XS 3153602 IC50 = 4470 nM T18664 C6W4XQ 3155531 IC50 > 500000 nM T18664 CVC41T 4526314 IC50 = 2690 nM T18664 C9WT3C 4737564 IC50 > 1000000 nM T18664 CP6DK4 5043631 IC50 > 1000000 nM T18664 CF2B7X 6442405 Ki > 100000 nM T18664 C5VP4M 6502047 IC50 > 500000 nM T18664 C1IP2G 7626526 IC50 = 100000 nM T18664 CH74YF 9112818 IC50 = 3019.95 nM T18664 C3CEP4 9841262 IC50 = 25000 nM T18664 C48MOV 9924775 IC50 = 20 nM T18664 C8XU2Z 10084259 IC50 = 18000 nM T18664 C5R6FZ 10130609 IC50 = 140 nM T18664 C6XJQ8 10398930 IC50 = 2140 nM T18664 CL6BN0 10406009 IC50 = 316.23 nM T18664 C2G6ER 11235803 IC50 ~ 11000 nM T18664 CKAW36 11338352 IC50 ~ 11000 nM T18664 C5MA2H 11362229 IC50 ~ 11000 nM T18664 CEZN60 11536404 IC50 = 436515.83 nM T18664 CYUF67 11560249 IC50 > 100000 nM T18664 C8UKO9 12351263 IC50 = 6456.54 nM T18664 CY3EL7 12639462 IC50 > 1000000 nM T18664 CNDB87 12675603 IC50 = 1995.26 nM T18664 C4T2NH 13059262 IC50 = 1550 nM T18664 C15IQF 13072144 IC50 = 141.25 nM T18664 CUVL56 13258570 IC50 = 630957.34 nM T18664 CF1EO5 14852550 IC50 = 890 nM T18664 C7OTE1 14906453 IC50 = 812.83 nM T18664 CQJ34A 15474479 IC50 = 7860 nM T18664 C8EAB7 15640477 IC50 = 102329.3 nM T18664 C31ZDL 17989764 IC50 = 3 nM T18664 CG4I3K 18184754 IC50 = 310 nM T18664 C1U0AG 18184758 IC50 = 91.2 nM T18664 CVZ4I8 18184779 IC50 = 110 nM T18664 C9KNO1 18417179 IC50 = 4680 nM T18664 CBYT29 18927006 IC50 = 660 nM T18664 C3VY6O 20110407 IC50 = 97723.72 nM T18664 CPLA13 20110740 IC50 > 1000000 nM T18664 C43EDK 20111303 IC50 > 1000000 nM T18664 C6AWZ9 21030535 IC50 = 3550 nM T18664 CMNR14 23725185 IC50 = 56.1 nM T18664 CBXC05 24424330 IC50 = 363 nM T18664 CH76FM 24458062 IC50 = 10 nM T18664 CB20PL 24795576 IC50 = 6 nM T18664 CVM48X 24894033 IC50 = 657000 nM T18664 CO1X6G 25017344 IC50 = 248.9 nM T18664 CL7AQ8 25017345 IC50 = 752.1 nM T18664 CWYO53 25017346 IC50 = 116.1 nM T18664 CAXI91 25017348 IC50 = 427.1 nM T18664 C5ZA4T 25017607 IC50 = 190.3 nM T18664 C5IXW8 25017608 IC50 = 383.1 nM T18664 CCKO19 25017611 IC50 > 5000 nM T18664 C0PE9N 25021166 IC50 = 347 nM T18664 C1RL0Z 25095848 IC50 = 4 nM T18664 C32ETF 25102032 IC50 = 8000 nM T18664 C5S7AV 25255635 IC50 = 1900 nM T18664 COG6B4 25561014 IC50 = 39 nM T18664 CH7K2U 41111610 IC50 > 100000 nM T18664 C9M2OV 42631278 IC50 = 133000 nM T18664 C2IUG6 42645607 IC50 = 8400 nM T18664 CL86VR 42645849 IC50 = 24000 nM T18664 CF0Q2G 42646079 IC50 = 12000 nM T18664 CJ97CU 42646080 IC50 = 4200 nM T18664 C9PTQ5 42646081 IC50 = 14000 nM T18664 CBI52J 42646085 IC50 = 2100 nM T18664 CQ2U6S 42646340 IC50 = 1000 nM T18664 C57DPZ 42646580 IC50 = 19000 nM T18664 CFO0G7 42646582 IC50 = 30000 nM T18664 C0CH9P 42646584 IC50 = 22000 nM T18664 C4E2LF 44128291 IC50 = 201.3 nM T18664 CRZ04P 44185045 IC50 = 1.698 nM T18664 C80SOB 44549116 IC50 = 4060 nM T18664 C80VGL 44549228 IC50 = 1840 nM T18664 CB62TJ 44549229 IC50 = 23300 nM T18664 CZ12LI 44549230 IC50 = 1862.09 nM T18664 C5XLF1 44549231 IC50 = 8510 nM T18664 CE0A4Y 44549232 IC50 = 14791.08 nM T18664 C1EKV9 44550621 IC50 = 269.15 nM T18664 C0F3PW 44550622 IC50 = 478.63 nM T18664 C3WSM8 44550737 IC50 = 6918.31 nM T18664 C04LIG 44550738 IC50 = 165.96 nM T18664 C42CZB 44550739 IC50 = 489.78 nM T18664 CV8X3S 44550740 IC50 = 5011.87 nM T18664 C08HAP 44550741 IC50 = 741.31 nM T18664 C26CPR 44550742 IC50 = 436.52 nM T18664 C56ISG 44550861 IC50 = 4073.8 nM T18664 CJ60RL 44550862 IC50 = 346.74 nM T18664 CU7L0S 44550864 IC50 = 95499.26 nM T18664 CS4CR5 44550865 IC50 = 218776.16 nM T18664 CL75VJ 44550866 IC50 = 19054.61 nM T18664 CWR2Z0 44550997 IC50 = 15488.17 nM T18664 CJM48I 44593853 IC50 = 0.9 nM T18664 C7K5ME 45140797 IC50 = 2300 nM T18664 CBCP74 45140975 IC50 = 18197.01 nM T18664 C4VUL3 45271579 IC50 = 17000 nM T18664 CCM9F4 45483976 IC50 = 930 nM T18664 CL4O9Q 45483983 IC50 = 2120 nM T18664 C6RPB1 45484093 IC50 = 1122.02 nM T18664 CDG80N 45484105 IC50 = 10471.29 nM T18664 CKW0V1 45591408 IC50 > 100000 nM T18664 C89VEA 45784884 IC50 = 194984.46 nM T18664 CJ2QP7 46831765 IC50 = 21 nM T18664 C2LP1G 46894146 IC50 = 354.81 nM T18664 C3V8TS 46933421 IC50 = 645654.23 nM T18664 CLAX29 46933424 IC50 = 489778.82 nM T18664 C5WES4 46933427 IC50 = 199526.23 nM T18664 CC9S7A 54761543 IC50 = 29 nM T18664 CALX42 56924669 IC50 = 4073.8 nM T18664 CPR2O8 56924670 IC50 = 2400 nM T18664 CX40EW 56950173 IC50 > 10000 nM T18664 C5TV9O 56950174 IC50 = 1800 nM T18664 C2BZ8E 56950175 IC50 = 6606.93 nM T18664 C59WSP 56950176 IC50 > 10000 nM T18664 C89HVZ 56950177 IC50 > 10000 nM T18664 CG83HI 56950178 IC50 = 1600 nM T18664 CANJ54 56950179 IC50 > 10000 nM T18664 C90WCO 56950316 IC50 = 12000 nM T18664 C38BSN 56950317 IC50 > 10000 nM T18664 CJE9X6 56950318 IC50 > 10000 nM T18664 CB4N0J 56950319 IC50 = 5100 nM T18664 CTX32Y 56950320 IC50 = 760 nM T18664 C72SOH 56950321 IC50 > 10000 nM T18664 C5KG3T 56950322 IC50 > 10000 nM T18664 CZWR80 56950453 IC50 = 15488.17 nM T18664 CP27FA 56950455 IC50 > 10000 nM T18664 CKF12Y 56950459 IC50 > 10000 nM T18664 CET81V 56950593 IC50 > 10000 nM T18664 C3NH9S 56950594 IC50 > 10000 nM T18664 C5FB4I 56950596 IC50 = 7585.78 nM T18664 CB98PJ 57394979 IC50 = 410 nM T18664 CU5ET1 57398502 IC50 = 275000 nM T18664 C4LO0S 57400169 IC50 = 67900 nM T18664 CI5CW0 59257514 IC50 = 130 nM T18664 CMJ1I9 60148506 IC50 = 154.88 nM T18664 C5NTI9 60165943 IC50 > 1000000 nM T18664 CRE8Q1 60165944 IC50 = 21877.62 nM T18664 COZ5D4 60165945 IC50 > 1000000 nM T18664 CR2QM7 60165946 IC50 > 1000000 nM T18664 CUF87Y 60165947 IC50 > 1000000 nM T18664 C3OHR5 60166095 IC50 > 1000000 nM T18664 CLBX87 60166096 IC50 = 95499.26 nM T18664 CTAR14 60166097 IC50 > 1000000 nM T18664 C7N9IK 60166098 IC50 > 1000000 nM T18664 C32VMN 60166099 IC50 = 69183.1 nM T18664 CI8SD2 60166100 IC50 > 1000000 nM T18664 CN04VS 60166227 IC50 > 1000000 nM T18664 CR15AG 60166228 IC50 = 7413.1 nM T18664 CDF5E1 60166229 IC50 = 1778.28 nM T18664 C81SRW 60166230 IC50 = 4265.8 nM T18664 CWTJ32 60166231 IC50 = 5128.61 nM T18664 CFN8T6 60166232 IC50 = 3715.35 nM T18664 CI1HK7 60166350 IC50 = 6025.6 nM T18664 C2F6XW 60166351 IC50 = 2187.76 nM T18664 C65QMZ 60166352 IC50 = 5370.32 nM T18664 C8ZI0R 60166353 IC50 = 7079.46 nM T18664 CASY70 60166475 IC50 = 5011.87 nM T18664 CCED97 60166476 IC50 = 7762.47 nM T18664 CRE1N7 60166477 IC50 = 1000 nM T18664 C0SY7C 60166478 IC50 = 831.76 nM T18664 CC0PD6 60166479 IC50 = 977.24 nM T18664 C6MTQ4 60166480 IC50 = 812.83 nM T18664 C4SN5T 60166610 IC50 = 1778.28 nM T18664 C51HFR 60166611 IC50 = 436.52 nM T18664 CU8MB7 66683014 IC50 = 8 nM T18664 C6MCT7 66683053 IC50 = 10 nM T18664 CNX2A7 69686440 IC50 > 10000 nM T18664 C91EJW 70148936 IC50 = 0.7 nM T18664 C5JP0T 71449674 IC50 = 141 nM T18664 C0I1PS 71449675 IC50 = 10471 nM T18664 CI0UW5 71449676 IC50 = 12 nM T18664 CV6A9Z 71451483 IC50 = 63 nM T18664 CZ0U6N 71451484 IC50 = 162 nM T18664 CB9QL5 71451485 IC50 = 8 nM T18664 C4Y9OB 71452048 IC50 = 156.2 nM T18664 C56IYB 71453311 IC50 = 0.54 nM T18664 C18XHL 71453312 IC50 = 19 nM T18664 C9WC7N 71453313 IC50 = 9 nM T18664 CI0E4J 71453314 IC50 = 676 nM T18664 CMQJ41 71453315 IC50 = 36 nM T18664 CU8WO4 71455022 IC50 = 23 nM T18664 CJ82PW 71455023 IC50 = 3 nM T18664 CK46JT 71455024 IC50 = 224 nM T18664 C2QO4D 71455025 IC50 = 372 nM T18664 CA2NQ0 71455026 IC50 = 62 nM T18664 CI0O2Z 71456811 IC50 = 234 nM T18664 C5R6FU 71456812 IC50 = 102 nM T18664 C90OBC 71456813 IC50 = 13 nM T18664 CRY48I 71458671 IC50 = 30 nM T18664 CS0DX3 71458672 IC50 = 20 nM T18664 C60IZO 71458673 IC50 = 2 nM T18664 C1Q9VE 71458674 IC50 = 324 nM T18664 CSXL15 71458675 IC50 = 7 nM T18664 CFIN48 71460495 IC50 = 33 nM T18664 C6VAY1 71460496 IC50 = 9 nM T18664 C2L0OM 71460497 IC50 = 32 nM T18664 CW0A2F 71460498 IC50 = 38 nM T18664 CW1GI7 71460499 IC50 = 33 nM T18664 CM3Q9Z 71460500 IC50 = 11 nM T18664 CG2L8T 71462206 IC50 = 71 nM T18664 CCN1Z0 71462207 IC50 = 955 nM T18664 CID4Z8 71462208 IC50 = 41 nM T18664 CL45WD 71575475 IC50 = 10300 nM T18664 CCRY62 71575476 IC50 = 98410 nM T18664 CB0M3U 71575478 IC50 = 18960 nM T18664 C5Y2NJ 71575575 IC50 = 56850 nM T18664 CD1L5A 71575576 IC50 = 121700 nM T18664 C8XW1K 71656212 IC50 = 3 nM T18664 CYO64A 71656315 IC50 = 12 nM T18664 CK1M6O 71656520 IC50 = 74 nM T18664 C4NW9M 71656525 IC50 = 6.9 nM T18664 C50OAM 71656796 IC50 = 270 nM T18664 C2TO5C 71656797 IC50 = 69 nM T18664 CN89IX 71656798 IC50 = 6 nM T18664 C49OFR 71656799 IC50 = 3 nM T18664 C92YGU 71657082 IC50 = 24 nM T18664 CV5PM2 71657185 IC50 = 18 nM T18664 CPT0H5 71657290 IC50 = 17 nM T18664 CM2ZB8 71657292 IC50 = 34 nM T18664 CBSW63 71657395 IC50 = 1100 nM T18664 CVUD47 71657398 IC50 = 98 nM T18664 C4IP1G 72197089 IC50 > 1000 nM T18664 C9EVP5 72197090 IC50 > 1000 nM T18664 CUAX51 72197091 IC50 > 1000 nM T18664 CWP34U 72197092 IC50 > 1000 nM T18664 CDN29K 72197093 IC50 = 346.5 nM T18664 CA9CX5 72197094 IC50 = 601.5 nM T18664 C5QGC9 72197264 IC50 = 250 nM T18664 C3C5FR 72197265 IC50 = 84.5 nM T18664 CO5Z4D 72197266 IC50 > 1000 nM T18664 CX1J5H 72197267 IC50 > 1000 nM T18664 CXS6H8 72197268 IC50 = 520.2 nM T18664 COMJ27 72197269 IC50 > 1000 nM T18664 CC95RF 72197270 IC50 > 1000 nM T18664 CSB3M1 72197441 IC50 = 170.9 nM T18664 CC26EQ 72197442 IC50 > 1000 nM T18664 C2HD9F 72197443 IC50 > 1000 nM T18664 CV9DU7 72197444 IC50 > 1000 nM T18664 C9F1KH 72197445 IC50 > 1000 nM T18664 C0KL4H 72197446 IC50 > 1000 nM T18664 CO9TL8 72197447 IC50 = 807.4 nM T18664 CJBN23 72197620 IC50 = 310 nM T18664 C7C3QK 72197621 IC50 = 16 nM T18664 CXQ9Y0 72197622 IC50 = 60 nM T18664 C4K7YM 72197623 IC50 = 28 nM T18664 CI54GL 72197627 IC50 = 49 nM T18664 CHF0K8 72197628 IC50 = 498.5 nM T18664 C5UT4O 72197629 IC50 = 27 nM T18664 CNB9D0 72197630 IC50 = 372.2 nM T18664 CT8LB2 72197631 IC50 = 98.1 nM T18664 COJ5V6 72197632 IC50 = 10 nM T18664 CVB7R8 72197633 IC50 = 209.4 nM T18664 CVUH81 72197634 IC50 = 137.2 nM T18664 CC1BN9 72197800 IC50 = 37 nM T18664 C9ZM3F 72197801 IC50 = 67 nM T18664 C8SC7B 72197802 IC50 = 190 nM T18664 C8GF3D 72197803 IC50 = 15 nM T18664 CF0XS6 72197804 IC50 = 6 nM T18664 CHV41T 72197805 IC50 = 15 nM T18664 CW29PH 72197806 IC50 = 28 nM T18664 C6W2NK 72197807 IC50 = 121.4 nM T18664 C9VGP6 72197808 IC50 = 139.2 nM T18664 C1Q5DT 72197809 IC50 = 334.9 nM T18664 CG2JM3 72197976 IC50 = 75 nM T18664 CSHI72 72197977 IC50 = 15 nM T18664 CMC2O6 72197978 IC50 = 48 nM T18664 C1NXE9 72197979 IC50 = 33 nM T18664 CVA0S1 72197980 IC50 = 23 nM T18664 CHYM43 72197981 IC50 = 12 nM T18664 C51DGL 72197982 IC50 = 140 nM T18664 CK5IH7 72198155 IC50 = 220 nM T18664 CM1Y2R 72198156 IC50 = 870 nM T18664 C3FW0E 72198160 IC50 = 36 nM T18664 CG9NE1 72198161 IC50 = 180 nM T18664 CUWA79 72198349 IC50 = 110 nM T18664 C10HES 72198350 IC50 = 370 nM T18664 CY46MV 72198351 IC50 = 650 nM T18664 CD51XB 72710925 IC50 = 4000 nM T18664 CTN8F6 72710929 IC50 = 338.84 nM T18664 CL57BZ 72710931 IC50 = 1300 nM T18664 C9Q5VB 72710932 IC50 = 1621.81 nM T18664 CZ62BF 72712915 IC50 = 398.11 nM T18664 CNHX60 72712916 IC50 = 251.19 nM T18664 CZI8Y2 72714182 IC50 = 2000 nM T18664 CTK95E 72714186 IC50 = 630 nM T18664 CJFH45 76308542 IC50 = 24547.09 nM T18664 C4FI6M 76313567 IC50 = 0.36 nM T18664 CD79KO 76319468 IC50 = 79432.82 nM T18664 C6H3KY 76323091 IC50 = 165958.69 nM T18664 CVR20B 76323092 IC50 > 1000000 nM T18664 C2J3DI 76330314 IC50 = 537031.8 nM T18664 CV8EW4 76333925 IC50 = 26302.68 nM T18664 C68NYM 76333926 IC50 = 75857.76 nM T18664 CMO84Z 88924517 IC50 > 10000 nM T18664 C2KHF7 89677087 IC50 = 3.5 nM T18664 CXT5C7 89682527 IC50 = 230 nM T18664 CPF01Q 89682653 IC50 = 28 nM T18664 CN8HX3 89682683 IC50 = 59 nM T18664 CY7PD2 89682704 IC50 = 5 nM T18664 CNU8L7 89682719 IC50 = 20 nM T18664 CAM63W 91827462 IC50 = 0.74 nM T18664 C6WMQ7 101885727 IC50 = 460 nM T18664 CO45UA 101885733 IC50 = 220 nM T18664 CL96MC 102532094 IC50 > 100 ug.mL-1 T18664 CFVX28 102596130 IC50 = 45.71 nM T18664 C41NLJ 117911680 IC50 > 10000 nM T18664 C9EU7M 118196651 IC50 = 5 nM T18664 CS5I8Y 118196675 IC50 = 3.6 nM T18664 CQ30UB 118196678 IC50 = 38 nM T18664 C1ICN5 118196759 IC50 = 8.9 nM T18664 C1VRX0 118196912 IC50 = 380 nM T18664 CP0CV7 118196917 IC50 = 9.2 nM T18664 CC3PB7 118679371 IC50 = 25 nM T18664 C4NV0G 118679372 IC50 = 41.9 nM T18664 C8S7ZV 118679375 IC50 = 22 nM T18664 CJC5B7 118679385 IC50 = 8.9 nM T18664 C1T4LJ 118679388 IC50 = 18.2 nM T18664 CEH2V7 118679411 IC50 = 72.8 nM T18664 CWS1R8 118679455 IC50 > 1000 nM T18664 CX17LN 118679456 IC50 = 10.6 nM T18664 CDN47F 118679473 IC50 > 1000 nM T18664 CAH0W8 118679482 IC50 = 21.7 nM T18664 CYA20V 118679490 IC50 > 1000 nM T18664 CC91ST 118679498 IC50 > 1000 nM T18664 CB54ZE 118721876 IC50 = 1.3 nM T18664 C84PJU 118721877 IC50 = 257 nM T18664 C61PQI 118721878 IC50 = 275 nM T18664 CE1PG3 118721879 IC50 = 131.83 nM T18664 C53PHK 118721880 IC50 = 1905 nM T18664 CJ60EQ 118721881 IC50 = 1659.59 nM T18664 CB0AT2 118721883 IC50 = 0.5495 nM T18664 CQ21VA 118721886 IC50 = 7.762 nM T18664 CO32MQ 118721887 IC50 = 5.495 nM T18664 CL9PU7 118721888 IC50 = 2818.38 nM T18664 CP9FN2 118721889 IC50 = 1122.02 nM T18664 CT6CE8 118721890 IC50 = 69.18 nM T18664 C87LMW 118721891 IC50 = 660 nM T18664 CD9V8S 118721892 IC50 = 42 nM T18664 C8UJ4Y 118721896 IC50 = 0.6918 nM T18664 CS91PZ 118727545 IC50 = 100000 nM T18664 CK9YC1 118727546 IC50 > 100000 nM T18664 CQ1MT5 118727547 IC50 > 100000 nM T18664 C6FP4M 118727548 IC50 > 100000 nM T18664 CSU24B 118727549 IC50 > 100000 nM T18664 CS15CM 118727550 IC50 > 100000 nM T18664 C3JVH2 118728497 IC50 = 208 nM T18664 CRZ8N5 118728498 IC50 = 98 nM T18664 CE3KF0 118729361 IC50 = 645.65 nM T18664 C3O2SZ 118729362 IC50 = 2570 nM T18664 CFTM51 118729369 IC50 = 47 nM T18664 C0M3VK 118729722 IC50 > 100 ug.mL-1 T18664 CBD8C5 118729723 IC50 > 100 ug.mL-1 T18664 CTX3W2 118729724 IC50 > 100 ug.mL-1 T18664 CP4D5Q 118729725 IC50 > 100 ug.mL-1 T18664 C0EA2W 118729726 IC50 > 100 ug.mL-1 T18664 CA2P3M 118729727 IC50 > 100 ug.mL-1 T18664 CUC21I 118729728 IC50 > 100 ug.mL-1 T18664 CWU09Y 118729729 IC50 > 100 ug.mL-1 T18664 CLV56Y 118729730 IC50 > 100 ug.mL-1 T18664 C8N5EQ 118729731 IC50 > 100 ug.mL-1 T18664 CH3C4J 118729732 IC50 > 100 ug.mL-1 T18664 C8A0KU 118736027 IC50 = 21000 nM T18664 C6Z3ME 118736028 IC50 = 83000 nM T18664 CCF89V 118736030 IC50 = 34000 nM T18664 C39SCH 118736201 IC50 = 49000 nM T18664 C94UVD 118736202 IC50 = 38000 nM T18664 CYZN76 122188783 IC50 = 3235.94 nM T18664 C0Y9DJ 122188784 IC50 = 7940 nM T18664 C78GBF 122189210 IC50 = 560 nM T18664 C32NYL 122189211 IC50 = 3230 nM T18664 CLHJ86 122189212 IC50 = 520 nM T18664 C7JU5Q 122530045 IC50 = 15 nM T18664 C52SOB 122653897 IC50 = 0.64 nM T18664 C25SVE 122653931 IC50 = 44 nM T18664 C21AXO 122653949 IC50 = 1.2 nM T18664 C59HJB 122653972 IC50 = 9.8 nM T18664 CG2V4P 122653979 IC50 = 6.5 nM T18664 CX9K8Z 122653997 IC50 = 2.2 nM T18664 C1IMT4 122654012 IC50 = 11 nM T18664 C3C8DJ 122654040 IC50 = 13 nM T18664 C06QVN 122654041 IC50 = 140 nM T18664 C39QXI 122654048 IC50 = 47 nM T18664 C3IG7K 122654166 IC50 = 2200 nM T18664 CA41RD 122654173 IC50 = 2000 nM T18664 CG95MA 122659523 IC50 = 53 nM T18664 CS9U3T 126502731 IC50 = 3 nM T18664 C0K3VD 127030391 IC50 = 31.2 nM T18664 CJ2DB9 127030392 IC50 = 1.41 nM T18664 COX84Q 127030393 IC50 > 10000 nM T18664 CBE5G6 127030394 IC50 = 97.5 nM T18664 C7EWF1 127032422 IC50 = 13.2 nM T18664 CM7DG0 127032456 IC50 = 104.4 nM T18664 CRDP70 127033069 IC50 = 376 nM T18664 CY13UL 127033070 IC50 = 10000 nM T18664 C6C3IR 127033071 IC50 > 10000 nM T18664 CBJF32 127034177 IC50 = 61.4 nM T18664 CEL8Z9 127034178 IC50 = 251.3 nM T18664 C92IQH 127034179 IC50 = 23.3 nM T18664 C46QDL 127034180 IC50 > 10000 nM T18664 CQ0YV3 127034181 IC50 > 10000 nM T18664 CB2AN6 127041070 IC50 = 11100 nM T18664 CU0D3S 130346049 IC50 = 4 nM T18664 CA47PL 132941103 IC50 = 840 nM T18664 CZ3F5D 135239539 IC50 = 11 nM T18664 CXP07U 136180342 IC50 = 34000 nM T18664 CU5DY3 136245185 IC50 = 524807.46 nM T18664 CT06QH 136961605 IC50 = 11000 nM T18664 C3P1UM 137349039 IC50 = 0.38 nM T18664 C0N8GW 137349224 IC50 = 46 nM T18664 C0U9TO 137546866 IC50 = 26 nM T18664 CH4Y5N 137632145 IC50 = 354 nM T18664 C1YI3Q 137633246 IC50 = 2000 nM T18664 CN4J0D 137633600 IC50 = 1500 nM T18664 CLSV56 137633822 IC50 = 1600 nM T18664 CY6M2X 137634001 IC50 = 1.9 nM T18664 CAY18O 137634472 IC50 = 132 nM T18664 CCYR94 137635253 IC50 = 24 nM T18664 CO5C8B 137635585 IC50 = 0.18 nM T18664 CV0K1Y 137637912 IC50 = 71000 nM T18664 C7Y1SZ 137637979 IC50 = 1100 nM T18664 C79RVX 137639265 IC50 = 4300 nM T18664 CNU07E 137640733 IC50 > 200000 nM T18664 C09GIF 137642130 IC50 = 890 nM T18664 C9M6CN 137644320 IC50 = 4700 nM T18664 C1RW8N 137644586 IC50 = 26 nM T18664 CHWY96 137644844 IC50 = 11000 nM T18664 CZ1EW2 137647242 IC50 = 1400 nM T18664 CWV12T 137647652 IC50 = 582 nM T18664 CSF8J7 137647975 IC50 = 6800 nM T18664 C7KJG5 137648574 IC50 = 3.2 nM T18664 CVA64G 137648891 IC50 = 0.3 nM T18664 CW5D8G 137649377 IC50 = 61000 nM T18664 CTP8G7 137650060 IC50 = 0.41 nM T18664 C80UIS 137650659 IC50 = 1 nM T18664 CPX0E7 137651000 IC50 = 3 nM T18664 C9HC8N 137651148 IC50 = 48000 nM T18664 CWZ92Q 137651267 IC50 = 390 nM T18664 CID71T 137652178 IC50 = 3200 nM T18664 CE7Z4T 137653761 IC50 = 1400 nM T18664 CGO57U 137653784 IC50 > 200000 nM T18664 C0OU2I 137653907 IC50 = 132000 nM T18664 CR26QT 137654372 IC50 = 2 nM T18664 CP40UN 137655811 IC50 = 242 nM T18664 C95ZXT 137656145 IC50 > 200000 nM T18664 C3JQ9D 137657257 IC50 > 200000 nM T18664 CDF0I3 137657433 IC50 = 12000 nM T18664 CGW6R8 137658312 IC50 = 39 nM T18664 CIZ61E 137658438 IC50 = 445 nM T18664 CQ2VL0 137659198 IC50 = 0.18 nM T18664 CGBW45 137659704 IC50 = 810 nM T18664 CZ90XQ 137659909 IC50 = 1.9 nM T18664 CCL26N 137662014 IC50 = 13000 nM T18664 CV90FH 137662219 IC50 = 1600 nM T18664 CYAI82 137662239 IC50 = 6 nM T18664 CB8IM1 138319671 Ki = 39 nM T18664 C5XM3H 145949852 IC50 > 10000 nM T18664 CSM7J0 145951205 IC50 > 10000 nM T18664 C4IX1W 145951504 IC50 > 10000 nM T18664 C06VUY 145951905 IC50 > 10000 nM T18664 CV0S3L 145953742 IC50 > 10000 nM T18664 C2KJ8F 145955689 IC50 > 10000 nM T18664 C46LCZ 145955918 IC50 > 10000 nM T18664 CP0L8K 145956576 IC50 > 10000 nM T18664 CEX3U4 145956825 IC50 > 10000 nM T18664 CX70KY 145957108 IC50 > 10000 nM T18664 CDEK59 145959588 IC50 > 10000 nM T18664 C09BZG 145965919 IC50 > 10000 nM T18664 CC5K7T 145966601 IC50 = 85 nM T18664 CMC75J 145967406 IC50 = 2200 nM T18664 CB0F4G 145968661 EC50 = 2800 nM T18664 CI30FS 145969336 IC50 = 13400 nM T18664 CX06IN 145969557 IC50 = 4500 nM T18664 CCU95Y 145969562 IC50 = 10500 nM T18664 CO21PR 145970662 IC50 = 6700 nM T18664 C94FEG 145970673 IC50 = 7900 nM T18664 CB4D5Q 145970899 IC50 = 11300 nM T18664 CTOF05 145971646 IC50 = 0.562 nM T18664 CDN40B 145972411 IC50 > 10000 nM T18664 CKT7O8 145977995 IC50 > 10000 nM T18664 CY34IF 145978111 IC50 > 10000 nM T18664 CL3O2T 145978936 IC50 = 1700 nM T18664 CQ9W6Y 145979178 IC50 = 1500 nM T18664 C1DOE8 145979233 IC50 = 70000 nM T18664 CUY93Q 145979773 IC50 = 770 nM T18664 CWG57U 145979792 IC50 = 910 nM T18664 CPR56F 145980320 IC50 = 25000 nM T18664 CVH06Z 145980369 IC50 = 1700 nM T18664 C7GVF2 145980839 IC50 = 30000 nM T18664 CGK3Z0 145981394 IC50 = 4800 nM T18664 CB4C0W 145981825 IC50 = 2400 nM T18664 CPQV82 145982453 IC50 = 69000 nM T18664 CCLU69 145984890 IC50 = 2000 nM T18664 CC9A5U 145986497 IC50 = 12000 nM T18664 CG3X5N 145986519 IC50 > 200000 nM T18664 CWZ54V 145986609 IC50 = 119000 nM T18664 CW8H9U 145986669 IC50 = 28000 nM T18664 CXK1L7 145987580 IC50 = 3300 nM T18664 CYK5R0 145987634 IC50 = 1000 nM T18664 CV1IH0 145988362 IC50 = 680 nM T18664 C1ZU6Q 145988983 IC50 > 200000 nM T18664 C03UND 145989088 IC50 = 1100 nM T18664 C48XSP 145989224 IC50 = 960 nM T18664 CJ39WH 145990024 IC50 = 2500 nM T18664 C4NGJ6 145990365 IC50 = 19000 nM T18664 C6HWO1 145990873 IC50 = 36000 nM T18664 C0ULZ5 145990999 IC50 = 710 nM T18664 C2RL1D 145991319 IC50 = 7200 nM T18664 CU20DV 145991376 IC50 = 18000 nM T18664 CL3GP7 145991606 IC50 = 36000 nM T18664 COTD15 145992359 IC50 = 20000 nM T18664 CK6IV0 145992600 IC50 = 5100 nM T18664 C5Q7TN 145993038 IC50 = 26000 nM T18664 CLIO86 145993082 IC50 = 1300 nM T18664 C9HKY2 145993604 IC50 = 5200 nM T18664 C6G5JR 145993738 IC50 = 53000 nM T18664 CB9QT5 145993762 IC50 = 16000 nM T18664 C1CI9P 145994066 IC50 = 34000 nM T18664 CNC0L1 155510621 IC50 > 1000 nM T18664 CEQ7G4 155510849 IC50 = 51 nM T18664 CC2JR4 155511252 IC50 > 1000 nM T18664 CCF96U 155511300 IC50 > 1000 nM T18664 CUDY82 155511307 IC50 = 138 nM T18664 C9CD3Q 155511585 IC50 = 11 nM T18664 CJ6IX3 155511908 IC50 = 136 nM T18664 C3HPT7 155512359 IC50 > 1000 nM T18664 C25OAR 155512542 IC50 = 2 nM T18664 C47JAI 155512548 IC50 = 29.6 nM T18664 CY3DO5 155512983 IC50 > 1000 nM T18664 CX98TQ 155513301 IC50 > 1000 nM T18664 CI2WL8 155513853 IC50 = 12 nM T18664 CY56UG 155514624 IC50 > 1000 nM T18664 CWH1J8 155515580 IC50 = 127 nM T18664 CVJE37 155515611 IC50 = 1100 nM T18664 C1RP4X 155517019 IC50 > 1000 nM T18664 CYQW63 155517808 IC50 > 10000 nM T18664 CHO79M 155520825 IC50 = 162 nM T18664 CBG4Q8 155521008 IC50 = 4 nM T18664 CV16WB 155522180 IC50 = 8700 nM T18664 C1TL7E 155523739 IC50 > 1000 nM T18664 CH3D1S 155524579 IC50 > 1000 nM T18664 CL6Z1R 155526799 IC50 = 510 nM T18664 CINM36 155526945 IC50 = 224 nM T18664 CB1X0F 155527149 IC50 > 1000 nM T18664 CV1N8B 155527481 IC50 = 67 nM T18664 CA6WY8 155529488 IC50 = 457 nM T18664 CHOD71 155530277 IC50 = 8.5 nM T18664 CAOX76 155531008 IC50 = 10200 nM T18664 C6Z9GK 155531741 IC50 = 262 nM T18664 C1S2BF 155531807 IC50 > 1000 nM T18664 C9KR3U 155532955 IC50 = 2400 nM T18664 CV2WL1 155533081 IC50 = 960 nM T18664 CP7Z6T 155533485 IC50 = 1300 nM T18664 CW7N6K 155533489 IC50 = 2 nM T18664 CUVQ19 155533981 IC50 > 1000 nM T18664 C9LG3S 155534745 IC50 > 1000 nM T18664 C3R4KU 155534895 IC50 > 1000 nM T18664 CGH7N2 155535470 IC50 = 3 nM T18664 CF5XG3 155535666 IC50 = 39 nM T18664 CQ94SW 155535689 IC50 = 424 nM T18664 C4OC2K 155536049 IC50 = 240 nM T18664 CA19JH 155536407 IC50 = 34 nM T18664 CU8V9J 155537287 IC50 = 194 nM T18664 CIJ5Q0 155537858 IC50 = 2200 nM T18664 C2MTW3 155538265 IC50 = 1000 nM T18664 CLXA98 155541762 IC50 > 1000 nM T18664 CQ8T0I 155542078 IC50 = 100 nM T18664 CQ67EK 155543660 IC50 = 2 nM T18664 C8XZ7V 155545255 IC50 = 51 nM T18664 CB96OD 155545265 IC50 = 2500 nM T18664 CL10QU 155545776 IC50 = 1300 nM T18664 C9WGK1 155547201 IC50 = 310 nM T18664 CFCX98 155547301 IC50 > 1000 nM T18664 C6TPM9 155549206 IC50 = 110 nM T18664 C5T2NH 155549374 IC50 = 389 nM T18664 CH78YM 155549832 IC50 = 9 nM T18664 C68KIQ 155550240 IC50 = 200 nM T18664 C4U9WO 155550747 IC50 = 17 nM T18664 CR0FM8 155551068 IC50 = 1000 nM T18664 CMS4Z6 155553816 IC50 = 5000 nM T18664 C0VW4R 155554535 IC50 = 89 nM T18664 CQN09X 155555471 IC50 = 5300 nM T18664 C9TMC2 155556133 IC50 = 2600 nM T18664 CSFQ35 155556385 IC50 > 1000 nM T18664 CQY53R 155557652 IC50 > 1000 nM T18664 CHZ68L 155558062 IC50 = 368 nM T18664 C8M2AD 155558440 IC50 > 1000 nM T18664 C6ZDW5 155560606 IC50 = 1400 nM T18664 CY52RZ 155560863 IC50 = 74 nM T18664 C9VPE4 155560882 IC50 > 1000 nM T18664 CB17KD 155561240 IC50 > 1000 nM T18664 CIUO47 155561644 IC50 > 1000 nM T18664 CXP2M5 155562137 IC50 > 1000 nM T18664 C3C2ZV 155562951 IC50 > 1000 nM T18664 CP43WE 155563376 IC50 > 1000 nM T18664 C50HVG 155566229 IC50 > 1000 nM T18664 CY40OE 155566729 IC50 = 12300 nM T18664 C0NQE3 155567474 IC50 = 8200 nM T18664 C0DVX5 155567982 IC50 > 1000 nM T18664 C0WQ7B 155568006 IC50 > 1000 nM T18664 CR18ZU 155568434 IC50 > 1000 nM T18664 C18FJS 155569023 IC50 = 1300 nM T18664 C6M8ET 155569148 IC50 = 250 nM T18664 D00NXA 2776266 IC50 = 100000 nM T18664 D02UVS 5455 IC50 = 977.24 nM T18664 D02ZQH 4362 IC50 = 16600 nM T18664 D03DXV 2739381 IC50 = 43000 nM T18664 D04BWH 2359 IC50 = 32000 nM T18664 D04DKX 7188 IC50 = 316.23 nM T18664 D05GPK 2734315 IC50 = 71000 nM T18664 D06BGU 44560666 IC50 = 817000 nM T18664 D07CER 45483984 IC50 = 790 nM T18664 D09OSN 151253 IC50 = 19000 nM T18664 D0A5OS 76765 IC50 = 2220 nM T18664 D0AR1Y 22022556 IC50 = 1700 nM T18664 D0C3JV 3690297 IC50 = 1950 nM T18664 D0F1BD 42797 IC50 = 1620 nM T18664 D0F1UD 4589192 IC50 = 7900 nM T18664 D0FD8G 6011033 IC50 = 31000 nM T18664 D0G0MZ 25021165 IC50 = 2 nM T18664 D0H6FG 10429254 IC50 = 25.12 nM T18664 D0I1WN 83648 IC50 = 2240 nM T18664 D0J8TY 5280436 IC50 = 6456.54 nM T18664 D0K9HO 25021164 IC50 = 140 nM T18664 D0O1UQ 2734389 IC50 = 20000 nM T18664 D0OD3U 2734388 IC50 = 38000 nM T18664 D0PC5A 44243144 IC50 = 22300 nM T18664 D0W1OX 10979337 IC50 = 10000 nM T18664 D0W7XR 11507802 IC50 = 54.4 nM T08133 D06UWF 121596688 IC50 = 14 nM T08133 C28QWT 17498 IC50 = 19100 nM T08133 C3YNP5 36060 IC50 = 159100 nM T08133 CSU9M6 346620 IC50 > 500000 nM T08133 CK0TE7 786338 IC50 = 1700 nM T08133 C6GKH2 11629903 IC50 = 37100 nM T08133 CZA48P 12982786 IC50 = 10800 nM T08133 C9MXF6 12987083 IC50 = 34900 nM T08133 C3NY9R 13144197 IC50 = 18600 nM T08133 CX0KW2 13317552 IC50 = 22000 nM T08133 CYU31X 16126768 IC50 = 12900 nM T08133 C7OI2D 16220361 IC50 = 20200 nM T08133 CRW4V2 60040027 IC50 = 14200 nM T08133 CXG28B 68577654 IC50 = 11300 nM T08133 CD0LU1 71659999 IC50 = 19800 nM T08133 CP7Y4F 71660000 IC50 = 18800 nM T08133 CC2FO4 71660002 IC50 = 18500 nM T08133 CNL1D4 71660004 IC50 = 28100 nM T08133 CG5M2U 71660030 IC50 = 93500 nM T08133 CJX3Z2 71660032 IC50 = 14400 nM T08133 C82TIK 71660034 IC50 > 500000 nM T08133 CY4F5M 71660035 IC50 = 412300 nM T08133 CHE90S 71660068 IC50 = 15000 nM T08133 C3ZL0J 71660069 IC50 = 16300 nM T08133 CT3H7S 71660071 IC50 = 89800 nM T08133 CEH53L 71660073 IC50 = 18800 nM T08133 CYK34Q 71660075 IC50 = 67900 nM T08133 CAP3K9 71660077 IC50 = 18900 nM T08133 CL5XH0 71660079 IC50 = 12100 nM T08133 C7TQH9 71660114 IC50 = 10000 nM T08133 C9UQ0S 71660116 IC50 = 9700 nM T08133 CN96XQ 71660117 IC50 = 9800 nM T08133 C24TOD 71660119 IC50 = 5200 nM T08133 C12FNQ 71660154 IC50 = 51300 nM T08133 CP9WS7 155289389 IC50 = 320 nM T08133 C2GIH9 155519330 IC50 = 600 nM T08133 CS7J2M 155561683 IC50 = 1700 nM T08133 D03TWR 596810 IC50 = 17700 nM T62306 D02YIZ 12560 EC50 = 50.12 nM T62306 D05SGO 16136567 EC50 = 0.03981 nM T62306 D05UYQ 15984937 EC50 = 12.59 nM T62306 D0LI1C 44469321 IC50 > 10000 nM T62306 C2YD7L 177964 IC50 = 3.981 nM T62306 C0Q6AD 9863611 EC50 = 1584.89 nM T62306 CT2PV5 9895192 IC50 = 338 nM T62306 CRVO02 10010118 EC50 = 0.047 nM T62306 CVN43M 11168753 Ki = 60 nM T62306 C6QC4T 11180385 Ki = 62 nM T62306 C8JY3R 11181688 EC50 = 0.22 nM T62306 CNR8W9 11192254 Ki = 255 nM T62306 C4PH2D 11203197 Ki = 78 nM T62306 CU85OX 11204067 Ki = 6 nM T62306 CO69KG 11215117 Ki > 10000 nM T62306 CB37MT 11226476 Ki = 55 nM T62306 CVSL74 11250008 Ki = 222 nM T62306 CWQS50 11341873 Ki = 8 nM T62306 CW8F3Z 11387240 EC50 > 10000 nM T62306 CP2RH4 11398651 Ki = 64 nM T62306 CMLB64 11398860 EC50 = 560 nM T62306 CH39JD 11408794 EC50 > 10000 nM T62306 C3CT8S 11410548 Ki = 16 nM T62306 CZ69KW 11433096 Ki = 8.3 nM T62306 C3GNM2 11444593 Ki = 11 nM T62306 CW69VS 11993730 EC50 = 10 nM T62306 C6UM8Q 11994554 IC50 = 74 nM T62306 C4H6TJ 11994555 Ki > 10000 nM T62306 CP10JO 11994556 Ki = 3566 nM T62306 CLT25A 11994557 Ki > 10000 nM T62306 CWD27T 11994558 Ki > 10000 nM T62306 C5M8NY 11994676 Ki > 10000 nM T62306 C8V2CB 11994677 Ki = 1389 nM T62306 CH2V4W 11994678 Ki = 335 nM T62306 C05LOR 11994679 Ki = 664 nM T62306 CUL1R2 11994680 Ki = 185 nM T62306 C5A6JO 11994798 Ki > 10000 nM T62306 CA3IL8 11994799 Ki > 10000 nM T62306 CK2AU6 11994800 Ki = 6064 nM T62306 C3FC1L 11994801 Ki > 10000 nM T62306 CN3XA5 11994802 Ki = 6064 nM T62306 CH0F1I 11994924 Ki = 701 nM T62306 CP1JT2 11994925 Ki = 57 nM T62306 CEI37D 11994926 Ki > 10000 nM T62306 CI2R3Y 11994927 Ki = 79 nM T62306 CKQ74V 11994928 Ki = 192 nM T62306 C4AS5F 11995040 Ki > 10000 nM T62306 CM02VW 11995041 Ki = 3237 nM T62306 CE0GN8 11995042 Ki = 2373 nM T62306 C13IDN 11995044 Ki > 10000 nM T62306 CY1PI8 11995045 Ki > 10000 nM T62306 C0KG2A 11995153 Ki = 196 nM T62306 C0OK9R 11995154 Ki = 4898 nM T62306 CBI1W2 11995155 Ki = 1524 nM T62306 CEAD80 11995156 Ki = 650 nM T62306 C58WXD 11995157 Ki = 2553 nM T62306 CLOV39 11995257 Ki > 10000 nM T62306 CFG24K 11995259 Ki = 9726 nM T62306 CNI15L 11995260 Ki > 10000 nM T62306 CR1TA3 11995261 Ki = 982 nM T62306 CI2F0X 11995356 Ki = 1197 nM T62306 CBV4Q8 11995357 Ki = 3247 nM T62306 CA37YG 11995358 Ki = 1486 nM T62306 CFR30Y 11995359 Ki = 1876 nM T62306 CW0X3E 11995454 Ki = 2777 nM T62306 C75LCF 12016400 IC50 = 2480 nM T62306 CXF80W 15604512 EC50 = 39.81 nM T62306 CU2LO6 15984134 EC50 = 19.95 nM T62306 CP1Y0C 15984238 EC50 = 50.12 nM T62306 CEY3H2 15984240 EC50 = 63.1 nM T62306 C46QET 15984241 EC50 = 25.12 nM T62306 C2VR7O 15984242 EC50 = 31.62 nM T62306 CMX86T 15984318 EC50 = 31.62 nM T62306 C5YH9J 15984938 EC50 = 10 nM T62306 C5PCN0 15984939 EC50 = 3.981 nM T62306 C20CRP 16040587 EC50 = 3.981 nM T62306 CPU95S 16040939 EC50 = 3.981 nM T62306 CJL7W4 16040940 EC50 = 6.31 nM T62306 C4RPF9 16040941 EC50 = 10 nM T62306 C0NXY5 16041119 EC50 = 1.995 nM T62306 C1HSE6 16041121 EC50 = 5.012 nM T62306 C8ZP3G 16041292 EC50 = 15.85 nM T62306 C2GXE4 16041481 EC50 = 19.95 nM T62306 CLV43P 16041483 EC50 = 50.12 nM T62306 C4AZ3J 16752689 EC50 = 10 nM T62306 C1R5ZT 23557214 IC50 = 228 nM T62306 C2RN1X 23557218 IC50 = 990 nM T62306 C5IF6D 23656869 IC50 = 2 nM T62306 CP3SQ6 25114744 Ki = 33 nM T62306 C71NBD 25114976 Ki = 62 nM T62306 CR4VP8 25114977 Ki = 18 nM T62306 CK9Q3J 25115200 Ki = 27 nM T62306 CRZL34 25115201 Ki = 51 nM T62306 CR2M4D 25115427 Ki = 87 nM T62306 CWT90D 25115428 Ki = 100 nM T62306 CLZ59N 25115429 Ki = 20 nM T62306 C50QRV 25115652 Ki = 17 nM T62306 C27GOD 25115653 Ki = 21 nM T62306 CM9KO5 25115654 Ki = 23 nM T62306 CV8IB0 44276703 IC50 = 169.82 nM T62306 C13JLQ 44292204 EC50 > 10000 nM T62306 C03ZUA 44292287 EC50 = 4200 nM T62306 CM1R3I 44292401 EC50 > 10000 nM T62306 C4QHT2 44292517 Ki = 2.7 nM T62306 CSP3V9 44380610 IC50 = 8.318 nM T62306 CK0C9G 44380651 IC50 = 15.14 nM T62306 CH2DY9 44380970 IC50 = 3.162 nM T62306 CMO6X0 44380971 IC50 = 7.586 nM T62306 C0IDK1 44412878 IC50 = 267 nM T62306 C9V7BW 44412894 IC50 = 52 nM T62306 C9DU5M 44417632 Ki > 10000 nM T62306 C13HKV 44417633 Ki = 6391 nM T62306 C4PG3H 44417740 Ki > 10000 nM T62306 CXV0Y3 44417743 Ki = 7295 nM T62306 C3E6VF 44417758 Ki > 10000 nM T62306 CP97WG 44432967 Ki = 889 nM T62306 C3AOB1 44432968 Ki = 342 nM T62306 CL7Y8O 44432969 Ki = 171 nM T62306 CH1TR0 44432970 Ki = 376 nM T62306 C5JM4E 44432971 Ki = 1946 nM T62306 C8XNS7 44432973 IC50 = 8 nM T62306 CWK83A 44432974 Ki = 31 nM T62306 CRXA72 44432975 IC50 = 3 nM T62306 CC02AP 44432976 Ki = 27 nM T62306 C5SUF3 44432977 Ki = 6 nM T62306 CG50ZB 44432978 Ki = 543 nM T62306 CF8Z7S 44432979 Ki = 41 nM T62306 CG8D5L 44432980 Ki = 57 nM T62306 C8Z0LX 44432981 Ki = 116 nM T62306 C7UDS1 44467360 Ki = 19000 nM T62306 CD31GV 44569919 EC50 = 630.96 nM T62306 CL34YF 44569920 EC50 = 794.33 nM T62306 CN92CB 44570013 EC50 = 2511.89 nM T62306 CJ75DW 44570112 EC50 = 1000 nM T62306 C78BLW 44570364 EC50 = 79.43 nM T62306 CQJ68M 44570365 EC50 = 31.62 nM T62306 C0SGW4 44570409 EC50 = 50.12 nM T62306 CR9YO2 44570410 EC50 = 79.43 nM T62306 C3QPK4 44570411 EC50 = 3.162 nM T62306 CJX16E 44570412 EC50 = 10 nM T62306 CKG64M 44570450 EC50 = 19.95 nM T62306 CR7AG3 44570451 EC50 = 251.19 nM T62306 CX8HP4 44570452 EC50 = 1000 nM T62306 CKON49 44570453 EC50 = 7.943 nM T62306 CPX08J 44570489 EC50 = 10 nM T62306 CE2BR6 44570490 EC50 = 63.1 nM T62306 CF13PE 44570491 EC50 = 5.012 nM T62306 C84ZAY 44570492 EC50 = 50.12 nM T62306 CM1L6X 44570527 EC50 = 2.512 nM T62306 CGB85R 44570528 EC50 = 63.1 nM T62306 C42PMN 44570529 EC50 > 10000 nM T62306 C5N2OP 44570567 EC50 > 10000 nM T62306 C08KZX 44570568 EC50 = 398.11 nM T62306 CP68WQ 44570608 EC50 = 2511.89 nM T62306 CA5ZR4 44571373 EC50 = 5011.87 nM T62306 CQ6PJ3 44571374 EC50 > 12589.25 nM T62306 C8V4TL 44571375 EC50 = 398.11 nM T62306 C89YAH 44571376 EC50 = 1584.89 nM T62306 C5DPW8 44571939 EC50 = 50.12 nM T62306 C2TC6J 44571940 EC50 = 5011.87 nM T62306 C7UCS4 44571989 EC50 = 501.19 nM T62306 C1TN7Q 44571990 EC50 = 1000 nM T62306 CJ72RL 44571991 EC50 = 630.96 nM T62306 CT3VL0 44572029 EC50 = 630.96 nM T62306 C7Q1VZ 44572030 EC50 = 794.33 nM T62306 CD36ZW 44572031 EC50 > 12589.25 nM T62306 C4HUN3 44572032 EC50 > 12589.25 nM T62306 CFM90N 44572090 EC50 > 12589.25 nM T62306 CUQ7Y5 44572091 EC50 > 12589.25 nM T62306 C5OY3E 44572092 EC50 = 3162.28 nM T62306 C5G3VM 44572093 EC50 > 3162.28 nM T62306 C0X8ML 44593551 EC50 = 251.19 nM T62306 C8SNQ9 44593552 EC50 = 398.11 nM T62306 CQI0D4 45102707 EC50 = 7.943 nM T62306 CSEP-69 45102708 EC50 = 6.31 nM T62306 CIGP20 46882302 EC50 = 199.53 nM T62306 CJG6E9 46882303 EC50 = 1995.26 nM T62306 CDF2Y1 46882304 EC50 > 12589.25 nM T62306 CNV0P8 46882347 EC50 > 2511.89 nM T62306 C37EWD 46882348 EC50 > 3162.28 nM T62306 C69AMR 46882349 EC50 = 501.19 nM T62306 CFZV45 46882350 EC50 = 2511.89 nM T62306 CSF43I 46882393 EC50 = 50.12 nM T62306 CB3QV6 46882394 EC50 = 7.943 nM T62306 C01GKH 46882395 EC50 = 3.162 nM T62306 CX7D3V 46882396 EC50 = 63.1 nM T62306 C7NWZ9 46882457 EC50 = 3162.28 nM T62306 C4BH9E 46882458 EC50 = 2.512 nM T62306 CJ50FM 46882459 EC50 > 12589.25 nM T62306 CJ69NR 46882460 EC50 = 2511.89 nM T62306 CERN34 46882461 EC50 = 7943.28 nM T62306 C3FA8G 46882519 EC50 = 794.33 nM T62306 CF8IJ2 46882520 EC50 = 39.81 nM T62306 CQN87I 46882521 EC50 = 10 nM T62306 C56ULO 46882522 EC50 = 3.981 nM T62306 CRZ95W 46882582 EC50 = 5.012 nM T62306 CX72IN 46882583 EC50 = 31.62 nM T62306 CSY8G1 46882623 EC50 = 1584.89 nM T62306 COW7N4 46882624 EC50 = 2511.89 nM T62306 C30RBS 46882625 EC50 = 2511.89 nM T62306 CM52FE 46882626 EC50 > 12589.25 nM T62306 CWCB97 46882627 EC50 > 12589.25 nM T62306 C16KTD 46882669 EC50 > 12589.25 nM T62306 CKJ2I6 46882670 EC50 > 12589.25 nM T62306 CHS14B 46882671 EC50 = 501.19 nM T62306 CK4ND8 46882672 EC50 = 125.89 nM T62306 C2OU8F 46882673 EC50 > 12589.25 nM T62306 CP84OR 46882710 EC50 = 3162.28 nM T62306 CPFM68 46882711 EC50 = 1258.93 nM T62306 CC05XO 46882712 EC50 = 19.95 nM T62306 CL3EI9 46882713 EC50 = 12.59 nM T62306 CZ15LN 46882714 EC50 = 25.12 nM T62306 CD24US 46882752 EC50 = 7.943 nM T62306 CAN69D 46882753 EC50 = 5.012 nM T62306 C0RQA4 46882754 EC50 = 158.49 nM T62306 CZ5N6R 46882755 EC50 = 1995.26 nM T62306 CBXT24 46882756 EC50 = 501.19 nM T62306 C39WEJ 46882794 EC50 = 158.49 nM T62306 CTJ41Q 46882795 EC50 = 39.81 nM T62306 C4OZ1U 46882796 EC50 = 63.1 nM T62306 CDK0Q3 46882797 EC50 = 19.95 nM T62306 C1RAX0 53322109 Ki = 3.4 nM T62306 C3CSX7 71720371 Ki = 2.63 nM T62306 CK1UL6 73353287 EC50 = 0.15 nM T62306 D03FQP 83954 IC50 = 3.388 nM T13863 C8VB4U 480183 Ki = 1160 nM T13863 CROX25 480185 Ki = 4390 nM T13863 C4S9WR 3000497 Ki = 5700 nM T13863 C4Z0XK 3010932 Ki = 5200 nM T13863 CM04US 20649518 IC50 > 500000 nM T13863 CA81RS 44144381 Ki > 10000 nM T13863 C4RSI0 46899736 Ki = 290 nM T13863 CX0Y2G 46899738 Ki > 10000 nM T13863 CAM3V7 50939649 Ki = 110 nM T13863 CHC74O 50939651 Ki = 2100 nM T13863 CA0G3M 57133681 IC50 > 500000 nM T13863 CN6CZ8 57154289 Ki = 88000 nM T13863 CV3M4L 71449633 Ki = 115000 nM T13863 CXT97V 71449635 IC50 > 500000 nM T13863 C28YUT 71451445 IC50 > 500000 nM T13863 CWQ5O0 71451447 IC50 > 500000 nM T13863 C30XPC 71453256 IC50 > 500000 nM T13863 CGM4Q1 71453258 IC50 > 500000 nM T13863 C5ZL0G 71453261 IC50 > 500000 nM T13863 C39ZJF 71453263 Ki = 82000 nM T13863 CV3T2M 71453265 IC50 > 500000 nM T13863 C5JKU3 71454986 IC50 > 500000 nM T13863 C2H9WA 71454988 Ki = 132000 nM T13863 CET86A 71454990 Ki = 187000 nM T13863 CQIB21 71456772 IC50 > 500000 nM T13863 CHNV94 71456774 IC50 > 500000 nM T13863 C3MT0E 71456776 IC50 > 500000 nM T13863 CXB02M 71458628 IC50 > 500000 nM T13863 CK7DL1 71458630 IC50 > 500000 nM T13863 CPJG15 71458632 IC50 > 500000 nM T13863 C51OSR 71458634 IC50 > 500000 nM T13863 CX37BW 71458636 IC50 > 500000 nM T13863 C04EON 71458638 Ki = 155000 nM T13863 CPDA60 71460459 IC50 > 500000 nM T13863 CC4P2V 71462161 IC50 > 500000 nM T13863 CU8WH5 71462163 IC50 > 500000 nM T13863 CK90PE 71462165 IC50 > 500000 nM T13863 CEXT02 71475974 Ki = 16300 nM T13863 C9TE8A 71475975 Ki = 27000 nM T13863 CI6FA7 71475976 Ki = 24000 nM T13863 C6E1GM 71475977 Ki = 12500 nM T13863 CLE0Y3 71476908 Ki = 65000 nM T13863 CAJ0C4 71476909 Ki = 50000 nM T13863 C5KQ9M 71476910 Ki = 64000 nM T13863 CUBF31 71477064 Ki = 148000 nM T13863 CRD18E 71477065 Ki = 196000 nM T13863 CHC7K2 71477066 Ki = 163000 nM T13863 CZH38E 71477067 Ki = 163000 nM T13863 CQT08V 71477068 Ki = 42000 nM T13863 C24WTK 71477222 IC50 > 500000 nM T13863 C1E0MZ 71477223 IC50 > 500000 nM T13863 C6CBP2 71477224 IC50 > 500000 nM T13863 CR47VE 71477225 Ki = 27000 nM T13863 CEA26W 71477226 IC50 > 500000 nM T13863 CSXC62 71477380 Ki = 137000 nM T13863 CE3LD8 71477381 Ki = 48000 nM T13863 CF67HS 71477382 Ki = 7600 nM T13863 CAOD57 71477383 Ki = 65000 nM T13863 CP7TO4 71477384 Ki = 70000 nM T13863 CT16CB 71477529 IC50 > 500000 nM T13863 CUC56G 71477530 IC50 > 500000 nM T13863 CN7IV2 71477531 IC50 > 500000 nM T13863 CQ7RZ1 71477532 IC50 > 500000 nM T13863 C4HPE8 71477533 IC50 > 500000 nM T13863 CIU9J6 71477683 IC50 > 500000 nM T13863 C3EOG6 71477684 IC50 > 500000 nM T13863 C5GKW9 71477685 Ki = 139000 nM T13863 CH3AO9 71477686 Ki = 207000 nM T13863 C5C4IM 71477687 Ki = 52000 nM T13863 CI5U2V 71477829 Ki = 208000 nM T13863 C2WGZ0 71477830 Ki = 217000 nM T13863 C15WQM 71477831 IC50 > 500000 nM T13863 CD8X3F 71477832 Ki = 22000 nM T13863 CSB35T 71477833 Ki = 19000 nM T13863 C1N4FS 71477979 Ki = 24000 nM T13863 C0H8NK 71477980 Ki = 10700 nM T13863 CPHV01 71477981 Ki = 8900 nM T13863 C6X5KL 71477982 Ki = 19000 nM T13863 C45FPN 71478120 Ki = 11800 nM T13863 CU2VL3 71478121 Ki = 40000 nM T13863 C4OGP2 71478122 Ki = 25300 nM T13863 C4IXP0 71478123 Ki = 40000 nM T13863 CVD3W9 71495381 Ki = 350 nM T13863 CNVH43 71495466 Ki = 400 nM T13863 CA5N2S 71495467 Ki = 750 nM T13863 CQ98NY 71495468 Ki = 3000 nM T13863 CE15GB 71495559 Ki = 10000 nM T13863 CW1Y2L 71495560 Ki = 3200 nM T13863 C5Q9BD 71495561 Ki = 3200 nM T13863 C36MRI 71495659 Ki = 770 nM T13863 C7PDA9 71495660 Ki = 310 nM T13863 CF3C8E 71495661 Ki = 210 nM T13863 CECD13 71495765 Ki = 1600 nM T13863 C7LXK1 71495766 Ki = 580 nM T13863 CKQ82B 71495974 Ki = 3300 nM T13863 CSV38K 71495975 Ki = 1300 nM T13863 C7QPA0 71495976 Ki = 3900 nM T13863 CI4P9Z 71495977 Ki = 2400 nM T13863 CE03BA 71496089 Ki = 790 nM T13863 CLO24G 71496201 Ki = 1300 nM T13863 CIE7A6 71496202 Ki = 1100 nM T13863 CAM0I4 71496204 Ki = 4400 nM T13863 CMC3L7 89399327 Ki = 1900 nM T13863 C1SAZ8 90666139 Ki = 1300 nM T13863 C2ERV8 90666140 Ki = 1200 nM T13863 CSO5R7 90666141 Ki = 460 nM T13863 C3F0PB 90666142 Ki = 1800 nM T13863 CG1W0R 90666143 Ki = 1300 nM T13863 CI3AX1 90666144 Ki = 180 nM T13863 C43YWM 90666145 Ki = 73 nM T13863 CT45NA 90666146 Ki = 1420 nM T13863 C56KQL 90666147 Ki = 940 nM T13863 CYUL31 118720337 Ki = 7.8 nM T13863 C4SUL9 118720338 Ki = 0.74 nM T13863 CP4F0X 118720339 Ki = 1.4 nM T13863 C0QI8C 118720340 Ki = 6.3 nM T13863 C6UG4N 118720341 Ki = 15.4 nM T13863 COFR38 118720342 Ki = 13.47 nM T13863 CA7O2K 118720343 Ki = 34.8 nM T13863 C3E7IH 118720344 Ki = 46.78 nM T13863 C9Z4AQ 118720345 Ki = 47.77 nM T13863 CKLU87 118720346 Ki = 24.84 nM T13863 C2NE9Q 118720347 Ki = 1.03 nM T13863 CS2G7Z 118720348 Ki = 2.56 nM T13863 CC2EV6 118720349 Ki = 1.98 nM T13863 CL28SC 118720350 Ki = 2.48 nM T13863 CF64QE 118720351 Ki = 20.79 nM T13863 C0IAV8 122182389 Ki = 3680 nM T13863 CXT84D 122182390 Ki = 1640 nM T13863 C6RDX4 122192767 Ki = 13600 nM T13863 CY0K9V 122192770 Ki = 19300 nM T13863 CP42JE 122192779 Ki = 81.9 nM T13863 C43TNZ 122192780 Ki = 87 nM T13863 C71IOQ 122192783 Ki = 546 nM T13863 CNJH01 122192784 Ki > 50000 nM T13863 C90LJI 127045142 Ki = 6230 nM T13863 CX52AQ 137631869 Ki = 5.3 nM T13863 CMB40N 137632239 Ki = 6 nM T13863 CDN14Z 137635697 Ki = 56 nM T13863 CV3I9R 137637849 Ki = 7 nM T13863 CI5VX9 137639355 Ki = 9 nM T13863 C5PHM2 137640910 Ki = 3.5 nM T13863 CI3JQ8 137640977 Ki = 5 nM T13863 C3TZH7 137640998 Ki = 5.3 nM T13863 CQ7N3P 137642872 Ki = 6 nM T13863 CVTM59 137644771 Ki = 5 nM T13863 CA7F3M 137645031 Ki = 3.1 nM T13863 C51JAT 137646077 Ki = 2.3 nM T13863 C94KVB 137646622 Ki = 690 nM T13863 C6G4RT 137647792 Ki = 13 nM T13863 C3P0CS 137648443 Ki = 340 nM T13863 C30ZQS 137648450 Ki = 5.2 nM T13863 CS03HK 137648571 Ki = 0.4 nM T13863 C6Z7LI 137653508 Ki = 1.1 nM T13863 CC0OE6 137653752 Ki = 6 nM T13863 C6HKV9 137654166 Ki = 1.74 nM T13863 CZW3F6 137655661 Ki = 560 nM T13863 CT6X1A 137657743 Ki = 1.2 nM T13863 C38KYF 137658118 Ki = 3.1 nM T13863 C0Z8RH 137658426 Ki = 2.6 nM T13863 CXEV32 137659374 Ki = 4 nM T13863 CAE43N 137659536 Ki = 5 nM T13863 C0SJX8 137661290 Ki = 1.5 nM T13863 CXZ3O7 137662143 Ki = 2.1 nM T13863 D07ZRG 46899577 Ki = 170 nM T13863 D08KCA 72429 Ki = 2400 nM T13863 D0W2SV 70689167 Ki = 3.3 nM T67163 C1EXW3 334509 EC50 = 26 nM T67163 CFQW02 9908426 EC50 = 3.9 nM T67163 CFQ46Z 11223729 EC50 = 31.9 nM T67163 C4WE3Y 20304994 EC50 = 4.1 nM T67163 CC9JB6 22015563 EC50 > 2000 nM T67163 CA6UK2 22015566 EC50 = 129.9 nM T67163 CWLP52 22015572 EC50 = 0.8 nM T67163 CR63DN 22015574 EC50 = 3.5 nM T67163 CJ16LU 22015582 EC50 > 2000 nM T67163 C7LJ9U 22015585 EC50 = 59.2 nM T67163 C1KQY0 24759785 EC50 = 218 nM T67163 CR7X1M 24856034 EC50 = 45 nM T67163 CC2K7Z 24856089 EC50 > 1000 nM T67163 C9F1UI 24856090 EC50 > 3000 nM T67163 CZ2IC7 44125335 EC50 > 1000 nM T67163 C8ZV1K 44125337 EC50 > 1000 nM T67163 CE5AI3 44125338 EC50 > 1000 nM T67163 CG74IY 44125340 EC50 > 1000 nM T67163 CP3JM2 44137900 EC50 > 1000 nM T67163 C21DXC 44137901 EC50 > 1000 nM T67163 CJA9S1 44137902 EC50 > 1000 nM T67163 CHB4G9 44231745 EC50 = 14 nM T67163 CK1U3D 44231857 EC50 = 38 nM T67163 C4KR1Y 44231980 EC50 > 1000 nM T67163 C41LNH 44231981 EC50 > 1000 nM T67163 CNS5Z9 44231982 EC50 > 1000 nM T67163 CWN5T1 44438317 EC50 = 113.1 nM T67163 CVD9B0 67046246 EC50 > 3000 nM T67163 CV04AZ 67046247 EC50 = 75 nM T67163 C9KOE6 67046278 EC50 > 3000 nM T67163 C91GSQ 67046282 EC50 > 3000 nM T67163 CIW78F 67046442 EC50 > 3000 nM T67163 CQ27LP 67140487 EC50 > 1000 nM T67163 CPOV75 67140847 EC50 = 25 nM T67163 CYDZ20 67265023 EC50 > 1000 nM T67163 C82BLR 68777542 EC50 > 1000 nM T67163 C89CQS 68779277 EC50 = 140 nM T67163 CND39E 68780103 EC50 > 1000 nM T67163 CB37TL 68781557 EC50 > 1000 nM T67163 C36CYH 68784863 EC50 > 1000 nM T67163 CGO8T6 135442495 EC50 = 77.5 nM T67163 C0L3EP 141243820 EC50 > 1000 nM T67163 CKL05J 155514632 EC50 > 1000 nM T67163 CB8Q5O 155518670 EC50 = 323 nM T67163 CGMO86 155524576 EC50 = 87 nM T67163 CXP1L7 155527972 EC50 > 3000 nM T67163 C7R8EZ 155532806 EC50 > 3000 nM T67163 CI32AK 155540265 EC50 > 3000 nM T67163 C8ZNC4 155551074 EC50 > 3000 nM T67163 C1N6JT 155551480 EC50 > 1000 nM T67163 C8E6RH 155552264 EC50 = 1585 nM T67163 C1CGJ7 155552765 EC50 > 3000 nM T67163 CK72EB 155553555 EC50 > 3000 nM T67163 CX7S9V 155556181 EC50 > 3000 nM T67163 CYN8B1 155556759 EC50 > 3000 nM T67163 C1TJY8 155557991 EC50 > 1000 nM T67163 C1QKZ9 155568991 EC50 > 3000 nM T29500 D00JVR 2267 Ki = 50.12 nM T29500 D01AZG 5073 Ki = 10 nM T29500 D01JUF 5775 Ki = 4.8 nM T29500 D03MIR 3157 Ki = 0.631 nM T29500 D04DKH 4418 Ki = 19.95 nM T29500 D04PHC 5816 EC50 = 75 nM T29500 D05MBZ 129211 EC50 = 0.13 nM T29500 D07MOX 439260 Ki = 20400 nM T29500 D08JIV 2162 Ki = 7943 nM T29500 D09EBS 4636 Ki = 831.76 nM T29500 D09MWJ 2092 Ki = 2.8 nM T29500 D0AE3X 2435 Ki = 5370.32 nM T29500 D0H3HM 60795 Ki = 100 nM T29500 D0H4JM 8969 Ki = 1.1 nM T29500 D0H7KF 5002 Ki = 100 nM T29500 D0O6IU 6041 EC50 = 0.86 nM T29500 D0O6IZ 4436 EC50 < 5011.87 nM T29500 D0P9RF 5401 EC50 = 0.5 nM T29500 D0U0VU 5312125 Ki = 19.95 nM T29500 D0V4QS 135398745 Ki = 1000 nM T29500 D0WV3U 4893 Ki = 0.21 nM T29500 D0Z1RV 135398737 Ki = 10 nM T29500 D05LGX 213041 Ki = 2089.3 nM T29500 D0N1HW 5311200 Ki = 2900 nM T29500 D00OWF 5280953 Ki > 10000 nM T29500 D00KZF 2419 Ki = 64.57 nM T29500 D01WJZ 60820 Ki = 47 nM T29500 D02FNU 56971 Ki = 220 nM T29500 D02LHR 33625 Ki = 25 nM T29500 D02ZSU 9838763 Ki = 11220.18 nM T29500 D03QMR 5685 Ki = 0.038 nM T29500 D04XCQ 10099811 Ki = 250 nM T29500 D05OVC 71310 Ki = 1949.84 nM T29500 D07BCO 5684 Ki = 66.07 nM T29500 D08OWQ 122295 Ki = 87 nM T29500 D0B1MJ 6918097 Ki = 25.12 nM T29500 D0B4TT 17747460 Ki = 31.62 nM T29500 D0L5TJ 10527469 Ki = 6.95 nM T29500 D0L9SN 4431 Ki = 0.96 nM T29500 D0N7LZ 126225 Ki = 19.95 nM T29500 D0P9FT 148842 Ki = 3.9 nM T29500 D0U3HP 164089 Ki = 0.08 nM T29500 D0YP7L 6604889 Ki < 10000 nM T29500 D0Z2UD 9872515 Ki = 79.43 nM T29500 D0Z3UP 216249 EC50 > 10000 nM T29500 CCO9N2 2894 Ki = 0.5888 nM T29500 C5H9CN 9287 Ki > 10000 nM T29500 C28VFY 60602 Ki = 25.01 nM T29500 CQ3R6M 72457 Ki = 1150 nM T29500 CN9GK1 104911 Ki = 322 nM T29500 CT1M8Y 119204 Ki = 3162.28 nM T29500 CFD09K 121102 Ki = 15.85 nM T29500 C2H1VA 131829 Ki = 4365.16 nM T29500 CY0O6P 151779 Ki = 147.91 nM T29500 CVA6M3 179268 Ki = 520 nM T29500 CZ0D8W 180707 Ki = 28 nM T29500 C28OMN 183528 Ki = 740 nM T29500 CF4V5Q 185076 Ki = 3311.31 nM T29500 CUO7A3 203096 Ki = 199.53 nM T29500 CHLI84 210172 Ki = 50.12 nM T29500 CE8AI0 456386 Ki = 170 nM T29500 C02ZTJ 456387 Ki = 130 nM T29500 CZN6S9 743974 IC50 > 39810.72 nM T29500 C1TV2F 1070749 Ki > 1200 nM T29500 CZG25W 1376848 Ki = 757 nM T29500 CAQ2J0 3034396 Ki = 4770 nM T29500 CU4T6Q 3086326 Ki = 10471.29 nM T29500 C2ZYB3 3826471 Ki = 91.2 nM T29500 CF6IK7 3894573 Ki = 15.85 nM T29500 CC9V5K 4013695 Ki = 1.82 nM T29500 C5K4PX 6603808 Ki = 72.44 nM T29500 C3A1FO 6604789 Ki < 10000 nM T29500 C0QCK1 6918455 Ki = 1995.26 nM T29500 CD0Z4I 6918648 Ki = 1995.26 nM T29500 CZ2M3Q 9794803 IC50 = 229.09 nM T29500 CD47WU 9795167 EC50 = 79.43 nM T29500 C2VS1K 9802999 Ki = 812.58 nM T29500 CN90IV 9804599 Ki = 100 nM T29500 C0L2CT 9808529 Ki > 2000 nM T29500 CG0I2Z 9816460 EC50 = 338.84 nM T29500 C4TKB3 9816461 EC50 < 100000 nM T29500 C0HZL7 9816515 EC50 = 50.12 nM T29500 C1XA0W 9816986 EC50 = 1995.26 nM T29500 C1X0UA 9817256 Ki = 4570.88 nM T29500 CO9VA3 9820671 IC50 > 1000 nM T29500 C2U3EZ 9822477 Ki = 193.29 nM T29500 CL2MG5 9822705 Ki = 15.84 nM T29500 CA2D7V 9822812 Ki = 79.62 nM T29500 CF0J1A 9822814 Ki = 7.95 nM T29500 C6JN8C 9822942 Ki = 43.35 nM T29500 C5DB6G 9823115 Ki = 17.01 nM T29500 CMB3R5 9824384 Ki = 0.07079 nM T29500 C6KJ7P 9827677 Ki = 100 nM T29500 CQZ6I0 9828476 Ki = 13.49 nM T29500 C0VO7E 9830292 Ki = 210 nM T29500 CHF96B 9837963 IC50 = 398.11 nM T29500 CCQ9W3 9838192 EC50 > 10000 nM T29500 C2EAU0 9838294 EC50 < 100000 nM T29500 C2O4HM 9838376 EC50 = 69.18 nM T29500 C3XCW9 9840212 EC50 < 100000 nM T29500 C8TE4O 9844321 Ki = 10.05 nM T29500 CAK7C9 9844511 Ki = 3915 nM T29500 C4YIM0 9845172 Ki = 37.57 nM T29500 C2TA1I 9845742 IC50 = 950 nM T29500 CXY3Z2 9847196 Ki = 1.86 nM T29500 C5I1XD 9847419 Ki = 221 nM T29500 CQM8A3 9847845 Ki = 3.7 nM T29500 CCB7Z6 9850782 Ki > 1658 nM T29500 CY2D5T 9851486 Ki = 263.03 nM T29500 C1SEL3 9859855 EC50 < 100000 nM T29500 CKF2T8 9864325 Ki = 62.62 nM T29500 CTY02P 9865254 Ki = 1400 nM T29500 C40JBW 9865801 Ki = 1.259 nM T29500 C1SOI8 9867138 Ki = 915.4 nM T29500 CAU0X5 9867616 Ki = 5.43 nM T29500 C7WAK9 9872440 Ki > 2000 nM T29500 CK5BJ6 9872851 Ki = 15.85 nM T29500 C7ER3F 9881853 EC50 < 100000 nM T29500 CV2HW7 9883506 Ki = 843 nM T29500 CTAC24 9885114 Ki = 787 nM T29500 CFW03P 9887458 Ki = 26.6 nM T29500 C6A9OS 9890459 Ki = 26310 nM T29500 C2SN0D 9891166 Ki = 4.47 nM T29500 CD2KC4 9891213 Ki = 0.1905 nM T29500 CQ9WG1 9891937 Ki = 79.43 nM T29500 CM7H6I 9891967 IC50 = 263.9 nM T29500 C3J8GU 9892409 Ki = 1995.26 nM T29500 CAY78Q 9892644 Ki = 47.54 nM T29500 CAM25C 9894665 Ki > 2000 nM T29500 C8HS4Q 9895326 Ki = 245.47 nM T29500 C5Y2AZ 9895338 Ki = 147.91 nM T29500 CK7C9L 9903313 EC50 = 251.19 nM T29500 C8RZ7N 9903932 EC50 < 100000 nM T29500 CYWQ50 9906447 Ki > 10000 nM T29500 C25XRA 9906677 Ki = 86.38 nM T29500 C7JFZ5 9906978 Ki = 41.7 nM T29500 CWV8K4 9908283 Ki = 119.18 nM T29500 CY2I0L 9908478 Ki = 5.88 nM T29500 C7SMT0 9908904 IC50 > 1000 nM T29500 CI1H6U 9909211 Ki = 12.59 nM T29500 CA0U4Y 9909471 Ki = 83.61 nM T29500 C0Y4CZ 9913449 Ki = 24 nM T29500 C78MDV 9913554 Ki = 1584.89 nM T29500 C5THY1 9913616 IC50 = 180.1 nM T29500 CBX74I 9915831 Ki > 2000 nM T29500 CT6QX7 9916549 Ki = 130 nM T29500 CCX3F8 9929277 Ki = 54.08 nM T29500 C7SOT8 9929936 Ki = 168.28 nM T29500 CUI0H7 9930376 IC50 = 560 nM T29500 C1C5KY 9931327 Ki = 380 nM T29500 C3L5MF 9932835 Ki = 52.89 nM T29500 CO2RS8 9934709 Ki = 1.288 nM T29500 C06OWM 9934955 IC50 = 3.2 nM T29500 CWO45F 9935387 Ki = 1000 nM T29500 CY8XG3 9938248 Ki = 78 nM T29500 CUQ8I5 9947861 EC50 = 61.66 nM T29500 C4G9VQ 9954092 Ki = 9.9 nM T29500 CFR41N 9957068 Ki < 5011.87 nM T29500 CBK3P7 9958160 Ki = 447.86 nM T29500 CD97EL 9959671 Ki = 190 nM T29500 C6LZS7 9959689 Ki = 250 nM T29500 CW89JP 9960311 Ki > 2000 nM T29500 CF1C5Q 9960497 Ki = 50 nM T29500 C7JXL1 9976756 Ki = 63.1 nM T29500 C2WVQ9 9982050 Ki = 15.2 nM T29500 CF7QK6 9982585 Ki = 360 nM T29500 C6PCS8 9984150 Ki = 1900 nM T29500 CD0IS5 9985476 Ki = 135 nM T29500 C4IG8L 10005161 Ki = 1.45 nM T29500 CA29FW 10015132 IC50 = 2041.74 nM T29500 C6XGV2 10020855 Ki = 53.1 nM T29500 CRH7V9 10026936 Ki = 900 nM T29500 CGN05I 10029146 Ki = 170 nM T29500 C05ICW 10031709 Ki = 250 nM T29500 C2EUY0 10035109 Ki > 10000 nM T29500 CZX09T 10038958 EC50 < 100000 nM T29500 C3A1ME 10047430 Ki = 4251 nM T29500 C9P4AC 10048729 Ki = 15.6 nM T29500 C71CVU 10060965 IC50 = 776.25 nM T29500 C0I2RV 10065903 Ki < 1000 nM T29500 CDF0Z2 10071710 Ki = 8.913 nM T29500 CN9B1F 10074286 Ki = 0.64 nM T29500 CVD98U 10083742 EC50 < 100000 nM T29500 CSW74O 10084685 EC50 < 100000 nM T29500 CC2ZY0 10089254 Ki = 199.53 nM T29500 C0IWD7 10091187 Ki = 43.3 nM T29500 C8NQ3I 10092649 Ki = 19 nM T29500 C4X0ID 10093481 Ki = 2.884 nM T29500 C3SJX0 10095044 Ki = 31.1 nM T29500 CP51OC 10097317 Ki = 570 nM T29500 CLW53J 10097792 Ki = 0.166 nM T29500 CE27RV 10135864 EC50 > 10000 nM T29500 C6FEY0 10151426 Ki = 66 nM T29500 COPD43 10160408 IC50 = 35.6 nM T29500 CSJ40T 10198532 EC50 = 1.585 nM T29500 CJ31LA 10199052 EC50 = 251.19 nM T29500 C7MKP9 10199335 Ki = 1318.26 nM T29500 CU2B9P 10221004 Ki = 912.01 nM T29500 CX9YD5 10221005 EC50 = 141.25 nM T29500 C12UXA 10221066 EC50 < 100000 nM T29500 CYR45Q 10227730 IC50 = 10000 nM T29500 CO64WJ 10236758 Ki = 776.25 nM T29500 CCF6U9 10244367 EC50 < 100000 nM T29500 C4Q2SH 10249573 Ki = 2511.89 nM T29500 C8SYA1 10252540 Ki = 0.1349 nM T29500 CBCZ21 10256583 Ki = 1.57 nM T29500 C9KDO8 10287924 Ki = 294 nM T29500 C0U3WR 10314056 Ki = 1294 nM T29500 C5VC9X 10317939 Ki > 1000 nM T29500 C62PAC 10318686 Ki = 2992 nM T29500 CJK89Q 10320782 Ki = 195.2 nM T29500 C3E5CB 10337773 Ki = 15848.93 nM T29500 C06YPQ 10342554 Ki = 1735 nM T29500 CIP38T 10344976 Ki = 1.072 nM T29500 C9IAV3 10346043 Ki > 1995.26 nM T29500 CI17PT 10348924 Ki = 6.5 nM T29500 COC7M0 10363912 Ki = 45.71 nM T29500 C0W8QR 10364538 Ki > 2000 nM T29500 C8GR5I 10364994 Ki = 0.537 nM T29500 C4RZL3 10368033 Ki = 35.1 nM T29500 CS7F3J 10371061 Ki = 220 nM T29500 CE9IN1 10378649 IC50 = 1949.84 nM T29500 C4H6YF 10379435 Ki = 1288.25 nM T29500 C3N7TF 10382537 Ki = 1905.46 nM T29500 CSAF82 10393665 Ki = 19 nM T29500 CG1IR6 10394346 Ki = 15.9 nM T29500 C0MBY3 10399043 IC50 = 162.18 nM T29500 C4TPN1 10413595 Ki = 1000 nM T29500 CQ52MH 10414908 Ki = 98 nM T29500 C7Z5FO 10415038 Ki = 24 nM T29500 C9EIT6 10415156 Ki = 610 nM T29500 CM76FU 10422033 EC50 < 5011.87 nM T29500 C0R3LA 10423384 EC50 < 100000 nM T29500 CP7B3M 10430193 Ki = 0.7413 nM T29500 CD7U5I 10433930 Ki > 3981.07 nM T29500 CCP0S9 10434440 Ki = 3.29 nM T29500 CIQ02H 10436842 Ki = 366 nM T29500 CZTU54 10437624 Ki = 240 nM T29500 CQ93PA 10438280 Ki = 45 nM T29500 CZH60T 10456471 Ki = 6.46 nM T29500 C7GEB0 10474042 Ki = 7.88 nM T29500 C5F7DM 10478121 Ki = 15.3 nM T29500 C0D1VZ 10479323 Ki = 8.913 nM T29500 CW16TJ 10481087 Ki = 280 nM T29500 C2T8JR 10503057 Ki = 3.33 nM T29500 CG3AW5 10504673 Ki = 0.33 nM T29500 C6UFO7 10506484 Ki = 490 nM T29500 C85BUY 10506673 Ki > 2000 nM T29500 CX73IB 10506729 Ki = 482 nM T29500 CY84UO 10507089 Ki > 2000 nM T29500 C69OVN 10507129 Ki = 77 nM T29500 CMG18U 10507220 Ki = 160 nM T29500 C3KX6O 10507357 Ki > 2000 nM T29500 C6C1NB 10507411 Ki = 500 nM T29500 CKJI08 10507500 Ki = 250 nM T29500 CJ0K1T 10507651 Ki = 380.19 nM T29500 C2U8AC 10508016 Ki = 138.04 nM T29500 C4XZ3Y 10508132 Ki = 1174.9 nM T29500 C0U9GR 10508330 Ki = 20 nM T29500 CZP09X 10508332 Ki = 162.18 nM T29500 C6M2OY 10526419 Ki = 29.1 nM T29500 C3O5XL 10527466 Ki = 0.84 nM T29500 CR0XV8 10530491 Ki > 2000 nM T29500 C35RPS 10530552 Ki = 16 nM T29500 C41XOR 10531022 Ki = 67 nM T29500 C0D4VW 10531157 Ki = 23 nM T29500 CE82ZX 10531476 Ki = 27 nM T29500 C4X9EF 10531532 Ki = 77.62 nM T29500 CJ3CL2 10531675 Ki = 36 nM T29500 C7MI2N 10531766 Ki = 223.87 nM T29500 C8PA4X 10549596 Ki = 2.754 nM T29500 CH8W9A 10554140 Ki = 7.5 nM T29500 CCKT30 10554745 Ki = 410 nM T29500 CPE27N 10554913 Ki = 8.4 nM T29500 C8NXE5 10554957 Ki = 400 nM T29500 C2ONS3 10555024 Ki = 490 nM T29500 CV7F9T 10555223 Ki = 1600 nM T29500 C16APC 10555288 Ki = 50 nM T29500 C7ROD9 10556164 Ki = 220 nM T29500 C2WGC8 10575494 Ki = 4.43 nM T29500 CQXU07 10575664 Ki = 8.56 nM T29500 CY04PF 10577609 Ki = 14.7 nM T29500 C7LWD8 10578548 Ki = 480 nM T29500 C93CLB 10578715 Ki = 361 nM T29500 C18HKX 10578735 Ki = 410 nM T29500 CT0ML5 10578926 Ki = 1500 nM T29500 C4SVP1 10578990 Ki = 1639 nM T29500 CF24MW 10579368 Ki = 977.24 nM T29500 C2LRK3 10579632 Ki = 27 nM T29500 CFQB52 10580182 Ki = 3130 nM T29500 C4L1WI 10582623 Ki = 8.2 nM T29500 CB2UE3 10582624 Ki = 12.59 nM T29500 CO23YX 10597140 Ki < 1000 nM T29500 CWM6C3 10599007 Ki = 21.08 nM T29500 CZ8IX1 10602912 Ki > 2000 nM T29500 CR8ZX2 10603727 Ki = 139 nM T29500 CD7W1O 10603739 Ki = 37 nM T29500 CK8SO7 10603951 Ki = 239.88 nM T29500 CX37LQ 10606657 Ki = 4.07 nM T29500 CZN59U 10606659 Ki = 61.2 nM T29500 COA7T4 10606661 Ki = 7.14 nM T29500 CY64KP 10606670 Ki = 3.31 nM T29500 C2G4IR 10617200 Ki = 46.77 nM T29500 CPI10N 10620533 Ki = 3.31 nM T29500 C9QT3I 10621309 Ki = 1.04 nM T29500 C8B5CJ 10621590 Ki = 79.43 nM T29500 CE5CU8 10621592 Ki = 446.68 nM T29500 CBH95U 10622156 Ki = 116 nM T29500 CNZU81 10622206 Ki = 63.1 nM T29500 C3XIF6 10622402 Ki = 0.74 nM T29500 CJ83IS 10622830 Ki = 95.2 nM T29500 CB4MC1 10624165 Ki = 2.31 nM T29500 CC34GW 10626453 Ki = 1700 nM T29500 CY4H5J 10626493 Ki = 72 nM T29500 COU08R 10626610 Ki = 250 nM T29500 C6BHD5 10626686 Ki > 2000 nM T29500 CNE1X0 10626726 Ki = 15 nM T29500 CUF48J 10626772 Ki = 310 nM T29500 CVG42P 10626843 Ki = 34 nM T29500 CQ13HM 10626910 Ki > 1750 nM T29500 CXD31C 10626911 Ki > 2000 nM T29500 CB26QH 10626982 Ki = 165.96 nM T29500 CYG6R7 10627003 Ki = 605 nM T29500 CSWC40 10627021 Ki = 269.15 nM T29500 CFA2R6 10627090 Ki = 130 nM T29500 C3TSO7 10627094 Ki = 430 nM T29500 CDC19N 10627155 Ki = 25 nM T29500 CF38IK 10627279 Ki = 100 nM T29500 CZ3T7S 10627329 Ki = 43 nM T29500 CER8L0 10640982 Ki = 1819.7 nM T29500 CS68CW 10643502 Ki = 2.58 nM T29500 CEP6D8 10644505 Ki = 2.11 nM T29500 CO7PA3 10647175 Ki = 1.64 nM T29500 C70QNW 10649481 Ki = 20 nM T29500 C9VY7F 10650129 Ki = 67 nM T29500 C6J4OK 10650633 Ki = 78 nM T29500 C4HP6A 10650726 Ki = 8.8 nM T29500 CLV1Q4 10650843 Ki = 606 nM T29500 CF1P6Z 10651080 Ki = 1174.9 nM T29500 CBN78H 10651219 Ki = 100 nM T29500 CV2HA5 10651636 Ki = 80 nM T29500 C3K7UP 10651654 Ki = 114.82 nM T29500 C07UGY 10673657 Ki = 130 nM T29500 CG6P7N 10674055 Ki = 255 nM T29500 C35NWA 10674133 Ki > 20000 nM T29500 CRQD91 10674333 Ki = 170 nM T29500 CX69JL 10674544 Ki = 1490 nM T29500 CQ9JN3 10674564 Ki = 465 nM T29500 C4EC8H 10674791 Ki = 48 nM T29500 C95VPX 10674840 Ki > 2000 nM T29500 CTB7L2 10674896 Ki = 151.36 nM T29500 CC8IT7 10675068 Ki = 150 nM T29500 C9KV5W 10678154 Ki = 1.01 nM T29500 C9TOQ8 10678161 Ki = 3.37 nM T29500 CBEP65 10688604 Ki = 93.33 nM T29500 CZL57G 10691912 Ki = 3.1 nM T29500 CG5CJ6 10692195 Ki = 1.63 nM T29500 C6ZLQ2 10693231 Ki = 1.56 nM T29500 CJ49EV 10694274 Ki = 191 nM T29500 CB0F2I 10697623 Ki = 440 nM T29500 CA80KS 10697912 Ki > 2000 nM T29500 C16NJO 10698141 Ki = 17 nM T29500 C6PVI9 10698570 Ki = 13 nM T29500 C4XZM6 10698974 Ki = 1940 nM T29500 CI4V5M 10699164 Ki = 15 nM T29500 C2OZ6W 10716964 Ki = 16.28 nM T29500 CR0QW8 10716965 Ki = 1.32 nM T29500 CN4P8H 10717073 Ki = 3.76 nM T29500 C0HO7D 10720893 Ki = 36 nM T29500 C87QBC 10721171 Ki = 140 nM T29500 C5WR2P 10721476 Ki = 400 nM T29500 C3WQ9B 10721564 Ki = 25 nM T29500 CZI63U 10721568 Ki > 2000 nM T29500 C5L4AS 10721730 Ki = 2820 nM T29500 CPF96G 10722045 Ki = 88 nM T29500 C6N7CQ 10722099 Ki = 58 nM T29500 CE2GK7 10739024 Ki = 25 nM T29500 CSN8Z1 10740369 Ki = 1.28 nM T29500 CLNP39 10740866 Ki = 2.27 nM T29500 CN8VP7 10741071 Ki = 0.92 nM T29500 CICD75 10742417 Ki = 9.27 nM T29500 C1QZ3O 10743042 Ki = 13.6 nM T29500 CD76GW 10743111 Ki = 11.3 nM T29500 CGQ8I3 10744391 Ki = 85 nM T29500 CU6HM4 10745305 Ki = 440 nM T29500 CHT1L0 10745380 Ki = 18 nM T29500 C1RZU6 10745566 Ki = 870 nM T29500 CA17HU 10745664 Ki = 150 nM T29500 CW91BJ 10745766 Ki = 100 nM T29500 C6IG0M 10745901 Ki = 49 nM T29500 CS3ON2 10746137 Ki = 730 nM T29500 CJ8VM0 10747021 Ki = 84 nM T29500 CBZP19 10747201 Ki = 130 nM T29500 CI5WL4 10763038 Ki = 1.16 nM T29500 C51YSW 10764133 Ki = 645.65 nM T29500 CFM65K 10767981 Ki = 0.9333 nM T29500 C0WMG4 10768610 Ki > 2000 nM T29500 C58CRB 10768829 Ki = 17 nM T29500 CV1JT2 10769037 Ki = 340 nM T29500 C63FIL 10769058 Ki = 410 nM T29500 CT1K3B 10769331 Ki = 41.69 nM T29500 C6JG4Z 10769621 Ki = 700 nM T29500 CV6T3C 10770007 Ki = 15 nM T29500 C8LZM3 10770057 Ki = 1225 nM T29500 C9ARF0 10770317 Ki > 2000 nM T29500 CS8QR2 10787126 Ki = 102.33 nM T29500 C8UB1S 10789770 Ki = 0.66 nM T29500 C1RC8F 10790988 Ki = 9.05 nM T29500 CMU59N 10791843 Ki = 320 nM T29500 C4XK8Y 10792591 Ki = 33 nM T29500 CS24OF 10792897 Ki > 1650 nM T29500 C6F5HP 10792898 Ki > 2000 nM T29500 CN71ZB 10793023 Ki = 110 nM T29500 C3O7YN 10793665 Ki = 123.03 nM T29500 CTXB06 10793720 Ki > 2000 nM T29500 C0D6MW 10793963 Ki = 64.57 nM T29500 CV39MC 10810527 Ki = 10.57 nM T29500 C6EWQ3 10811627 Ki > 5000 nM T29500 CHIR21 10812130 Ki = 0.66 nM T29500 CXU6D7 10815549 Ki = 93 nM T29500 CN6ZP7 10815593 Ki = 53 nM T29500 C4ZNR1 10816815 Ki = 310 nM T29500 C68UVF 10816832 Ki = 810 nM T29500 CO73GU 10816903 Ki = 510 nM T29500 CID39T 10817365 Ki = 30 nM T29500 CBO8N9 10818003 Ki = 162.18 nM T29500 CFC95U 10834793 Ki = 2.399 nM T29500 C8MHZ9 10835110 Ki = 1995.26 nM T29500 C5NFU1 10836245 Ki = 413 nM T29500 CIY58E 10839105 Ki = 120 nM T29500 CKS74R 10839106 Ki = 110 nM T29500 C5SC1X 10839825 Ki = 1100 nM T29500 CP78AK 10840177 Ki = 270 nM T29500 C49YSD 10840781 Ki = 1300 nM T29500 C4LV0H 10841070 Ki = 100 nM T29500 CE80NV 10841190 Ki = 204.17 nM T29500 C2RXD0 10841296 Ki = 320 nM T29500 CYSL64 10841387 Ki = 416 nM T29500 C8TED5 10841819 Ki = 2630 nM T29500 CO9WP2 10841851 Ki = 720 nM T29500 CI9UL7 10844296 Ki = 2.71 nM T29500 C3Z6PT 10874628 IC50 > 30000 nM T29500 C70LSM 10880840 Ki = 977.24 nM T29500 C3I1CT 10892762 Ki = 332 nM T29500 CEUD36 10893672 Ki = 33.13 nM T29500 CKYE37 10895266 Ki = 4073.8 nM T29500 CB1HW4 10905809 IC50 > 30000 nM T29500 C8VT6G 10916464 Ki = 645.65 nM T29500 CBH30I 10916771 Ki = 2.01 nM T29500 C2YHI8 10917023 Ki = 26.92 nM T29500 CD7QW2 10917316 Ki = 8.04 nM T29500 CH95TI 10923927 Ki = 2137.96 nM T29500 C1UZ3L 10928121 Ki < 10000 nM T29500 C4GCP7 10928161 Ki = 9549.93 nM T29500 C0N6KJ 10928520 Ki = 1.76 nM T29500 CMK6P8 10928757 IC50 > 30000 nM T29500 C3CI6Z 10934575 EC50 = 0.4169 nM T29500 CTO4Z9 10949698 Ki = 53.39 nM T29500 C5E8MI 10950119 Ki = 14.45 nM T29500 CAIJ61 10961351 Ki = 3.77 nM T29500 CW6T1N 10971791 Ki = 20.89 nM T29500 CH0VN7 10972370 IC50 > 30000 nM T29500 CIU42D 10973463 IC50 > 30000 nM T29500 CX5M6J 10974101 Ki = 4.7 nM T29500 CUK3X0 10982853 Ki = 55 nM T29500 CM5Y6J 10994432 IC50 = 6800 nM T29500 C4VA7K 10994660 IC50 > 30000 nM T29500 CC2NG9 10994812 Ki = 1.44 nM T29500 C8AG4Z 11005226 IC50 > 30000 nM T29500 C2BF0W 11014848 Ki = 49.84 nM T29500 CFO15P 11015356 IC50 = 1560 nM T29500 CD4LJ1 11027118 IC50 = 26900 nM T29500 CGW87Y 11034737 EC50 = 6.026 nM T29500 CZM27Y 11039289 Ki = 1.2 nM T29500 CH9O0P 11046644 Ki = 4.21 nM T29500 C10SEU 11047971 Ki < 10000 nM T29500 C48QYR 11058166 Ki = 380.19 nM T29500 CQ61ZR 11059085 IC50 > 30000 nM T29500 C7JI1M 11059195 Ki < 10000 nM T29500 C8L9KE 11059896 IC50 = 7000 nM T29500 C7R2AZ 11079593 Ki = 512.86 nM T29500 CUZ38C 11081136 Ki = 2.01 nM T29500 C91BKL 11090351 Ki = 2290.87 nM T29500 CF32NC 11092254 Ki = 3.95 nM T29500 CFE1M7 11097789 EC50 = 6.026 nM T29500 CTG4I5 11098175 EC50 = 3.631 nM T29500 C9CUO6 11102065 IC50 = 7900 nM T29500 CB7GA9 11102302 Ki = 2041.74 nM T29500 C84VUJ 11108001 EC50 = 1.995 nM T29500 CR6K4V 11109088 EC50 = 0.5012 nM T29500 C9ULK0 11112527 Ki = 61.66 nM T29500 CANW92 11112933 IC50 > 30000 nM T29500 CJT65Y 11123606 Ki = 20.28 nM T29500 CF68CS 11133288 Ki = 2.818 nM T29500 C7MD3R 11133868 Ki = 27.54 nM T29500 C3ZJK1 11134424 Ki = 0.75 nM T29500 CC0HY8 11135150 Ki = 75.86 nM T29500 CG40BP 11140345 EC50 = 85.11 nM T29500 CO0XW1 11140347 EC50 = 1.862 nM T29500 CA7Y5Z 11144555 Ki = 5.51 nM T29500 CSX94J 11144809 Ki = 100000 nM T29500 C73DFT 11145007 Ki = 49.08 nM T29500 CUNH28 11152823 Ki = 79.43 nM T29500 C0W4OI 11154198 Ki = 4.97 nM T29500 C7VKQ5 11164948 Ki = 295.12 nM T29500 CUE3X2 11176459 Ki = 46.18 nM T29500 C0UQ5K 11191047 Ki = 262.76 nM T29500 CCX87L 11200086 Ki = 7.76 nM T29500 C4DUK6 11201573 Ki > 1000 nM T29500 C4J8YG 11211017 Ki = 255 nM T29500 CO58DX 11224478 Ki > 1000 nM T29500 CR10CS 11234230 Ki = 35.94 nM T29500 CKEJ43 11270912 Ki = 5.38 nM T29500 C90UKI 11281005 Ki = 575.44 nM T29500 CR2DJ1 11282574 Ki = 7.413 nM T29500 C1VNU0 11303180 Ki = 131.95 nM T29500 CE03YG 11303253 Ki = 54.99 nM T29500 CO6NX8 11315660 Ki = 57.65 nM T29500 CCQ0S5 11338016 Ki = 12.3 nM T29500 CT3V5I 11338314 Ki = 1100 nM T29500 CG93PV 11348796 Ki = 274.38 nM T29500 CTB03C 11372228 Ki = 20.25 nM T29500 CJQ71D 11384983 Ki = 122.03 nM T29500 CZ2GN9 11394353 Ki = 84.08 nM T29500 CJLS45 11395842 Ki = 127.8 nM T29500 C7KX6F 11430126 Ki = 0.537 nM T29500 C7EVT0 11430491 Ki = 0.309 nM T29500 C7QX9L 11431037 Ki = 790.88 nM T29500 C9BNX8 11440979 Ki > 1000 nM T29500 CM8I7N 11454386 Ki = 1.259 nM T29500 C89FRU 11464777 Ki = 13.11 nM T29500 C6OVE5 11474152 Ki = 73.53 nM T29500 C6UBN9 11474937 Ki = 35.56 nM T29500 C51OVT 11485631 Ki = 8.21 nM T29500 C8Q1LZ 11486511 Ki = 11.5 nM T29500 C3NF7L 11487449 Ki = 13.61 nM T29500 C8TDA7 11488170 Ki = 39.81 nM T29500 CTMH12 11505007 Ki = 39 nM T29500 CS20NG 11519153 Ki = 133 nM T29500 CI8GN0 11532563 Ki = 1.995 nM T29500 C0MF3O 11539392 Ki = 0.7943 nM T29500 COC6U3 11554541 Ki = 0.3981 nM T29500 C2IE4D 11583392 Ki = 1 nM T29500 C6D1MA 11584660 Ki > 1995.26 nM T29500 CJW9E6 11604548 Ki = 0.2512 nM T29500 C6JRN0 11619713 Ki = 2.512 nM T29500 C3IHP8 11626704 Ki = 0.1585 nM T29500 C9VAI5 11633517 Ki = 0.2512 nM T29500 CL6XP8 11638677 Ki = 5.248 nM T29500 CZA0M9 11653915 Ki = 102.8 nM T29500 C9I7KB 11669646 Ki = 0.3981 nM T29500 CUVL17 11705133 Ki = 6.31 nM T29500 C7RAS6 11712250 Ki = 0.5623 nM T29500 C7PK3H 11712470 Ki = 0.7943 nM T29500 CIFM13 11729700 Ki = 245.47 nM T29500 CL8HU6 11730709 IC50 = 9500 nM T29500 CR1L6N 11732516 Ki = 258.92 nM T29500 C12YTV 11742585 Ki > 2000 nM T29500 CJ60OP 11742834 Ki = 0.03981 nM T29500 C3G4FS 11751173 Ki = 0.6761 nM T29500 CO50RT 11757736 Ki = 440 nM T29500 CA9XK6 11761245 Ki = 13.8 nM T29500 C06HZD 11782656 Ki = 270 nM T29500 C28UNM 11784634 Ki = 218.78 nM T29500 C4VL6W 11801214 Ki > 2000 nM T29500 CFTI34 11801828 Ki = 1778.28 nM T29500 C4ZXG0 11801861 Ki = 15500 nM T29500 C2RPQ0 11802456 Ki = 32 nM T29500 C1VWL5 11811395 Ki = 1000 nM T29500 C1H3FR 11812340 Ki = 27.54 nM T29500 C3XOR7 11825888 Ki = 162.18 nM T29500 C79MQD 11826825 IC50 > 30000 nM T29500 CUB53N 11857638 Ki = 144 nM T29500 C29HBR 11857639 Ki = 470 nM T29500 C29FMG 11857709 Ki = 123 nM T29500 CX50UR 11857710 Ki = 82 nM T29500 CW6V5E 11857711 Ki = 107 nM T29500 CD50HW 11857791 Ki = 91 nM T29500 CGL5D9 11857792 Ki = 216 nM T29500 CE0U9G 11857793 Ki = 181 nM T29500 CYJ5I7 11857794 Ki = 261 nM T29500 C9S5NU 11857861 Ki = 354 nM T29500 CU83FA 11857862 Ki = 278 nM T29500 CUO32E 11857863 Ki = 639 nM T29500 CD7O6J 11857864 Ki = 299 nM T29500 CXLW54 11948707 Ki = 378 nM T29500 C8JQL7 11957735 IC50 > 10000 nM T29500 CH1WZ3 11984570 Ki = 18 nM T29500 CJP2T4 11994550 Ki = 48.98 nM T29500 CHE4O6 11994665 Ki = 17.78 nM T29500 C0ZRF5 11994667 Ki = 10.96 nM T29500 CQW63S 11994668 Ki = 61.66 nM T29500 CVNL73 11994670 Ki = 549.54 nM T29500 C1BZQ0 11994673 Ki = 371.54 nM T29500 CB3DJ5 11994797 Ki = 19.05 nM T29500 C1KQO2 11994915 Ki = 186.21 nM T29500 CU17YO 11995033 Ki = 151.36 nM T29500 C3F1BT 11995035 Ki = 549.54 nM T29500 C1A2IB 12001199 Ki < 794.33 nM T29500 C8W5JG 12039032 Ki = 10000 nM T29500 CY8DS2 12134985 Ki > 10000 nM T29500 C4CI5P 12134986 Ki = 4456 nM T29500 CS6BU1 12134987 Ki > 10000 nM T29500 CPX75G 12134991 Ki > 5000 nM T29500 CI52SU 12134994 Ki = 1878 nM T29500 C8WEX1 12134995 Ki = 1063 nM T29500 C6S9BY 12134996 Ki > 5000 nM T29500 C2U3RT 12764879 EC50 > 10000 nM T29500 C0B1QO 12764880 EC50 > 10000 nM T29500 CFN31J 12840734 Ki = 264.47 nM T29500 C6P7TB 12840735 Ki = 220.52 nM T29500 C2V9FL 13091268 Ki = 42.7 nM T29500 CMA46J 13305910 Ki = 5.754 nM T29500 CN2ZQ5 13911290 Ki = 1.22 nM T29500 CV08GM 14378574 Ki = 360 nM T29500 C4E7NH 14423371 Ki = 0.1096 nM T29500 CMO81H 14925759 Ki = 74.13 nM T29500 CKVQ30 15054191 Ki = 2.57 nM T29500 C8BF2P 15254720 Ki = 10 nM T29500 C2OEA5 15480820 Ki = 11.75 nM T29500 CQ5ZJ2 15546405 Ki = 10000 nM T29500 C1CX2S 15675860 Ki < 100000 nM T29500 CRTO23 15840661 Ki = 125.89 nM T29500 CPR25X 15986917 Ki < 2511.89 nM T29500 C5KW3L 15987108 Ki < 794.33 nM T29500 CT03WI 16040907 Ki = 107 nM T29500 CW5NS1 16041090 Ki = 214 nM T29500 C03VCW 16041091 Ki = 69 nM T29500 CM3O4Z 16041092 Ki = 60 nM T29500 CUL5M9 16041263 Ki = 39 nM T29500 C6S8AM 16041264 Ki = 71 nM T29500 CYTD80 16041265 Ki = 50 nM T29500 C86MYV 16041449 Ki = 112 nM T29500 CHF7K6 16041451 Ki = 81 nM T29500 CCJ65Y 16041628 Ki = 76 nM T29500 CE2Z7Y 16041629 Ki = 36.4 nM T29500 CRJX49 16041630 Ki = 36 nM T29500 CDTN28 16121006 Ki = 15.85 nM T29500 CERP08 16219807 Ki < 10000 nM T29500 CZ2IS9 16660294 Ki > 10000 nM T29500 CZ8S6B 16721032 Ki = 0.871 nM T29500 C7KS8E 16721110 Ki = 4.467 nM T29500 C3GD2P 17753379 Ki = 78 nM T29500 CM60NI 17804479 EC50 = 791 nM T29500 CN0CH5 18187410 Ki = 3 nM T29500 CT3OK4 18738380 Ki = 10000 nM T29500 CF1DM9 18738384 Ki = 615 nM T29500 CEP14V 18738385 Ki = 384 nM T29500 CM6YI0 18738386 Ki = 259 nM T29500 CCO79B 18738387 Ki > 5000 nM T29500 C9E4ID 18738412 Ki = 3719 nM T29500 C2YEK1 19063108 IC50 = 206 nM T29500 CYT58A 19085820 Ki = 133 nM T29500 CHM64Z 19085827 Ki = 1650 nM T29500 CV8X0D 19085829 Ki = 50 nM T29500 C9CL0I 19085832 Ki = 108 nM T29500 C2EYW8 19085836 Ki = 1152 nM T29500 C6KSV0 19085839 Ki = 301 nM T29500 CRU75T 19085858 Ki = 10 nM T29500 CN5XJ1 19085866 Ki = 14 nM T29500 C2L1IX 19085869 Ki = 37 nM T29500 C4V1LT 19085876 Ki = 7.3 nM T29500 C7A2EC 19085881 Ki = 75 nM T29500 C8RDC1 19085894 Ki = 6.8 nM T29500 CC1Y7N 19085914 Ki = 15 nM T29500 C7T6HA 19085921 Ki = 1958 nM T29500 C7M9NZ 19085926 Ki = 20 nM T29500 CPJG69 20215436 Ki = 0.46 nM T29500 C4GM9S 20750645 Ki > 5000 nM T29500 C3T5HF 21509921 Ki = 3162.28 nM T29500 CD9Y0E 21712258 Ki > 2000 nM T29500 CT7XG9 21830793 Ki > 10000 nM T29500 C21LHM 22493224 EC50 = 199.53 nM T29500 C4UYD5 22493225 EC50 < 5011.87 nM T29500 C9V4MO 22493231 EC50 = 79.43 nM T29500 CKB2N6 22493233 EC50 < 100000 nM T29500 C0P2UY 22493236 EC50 = 5.012 nM T29500 C02AEX 22493245 Ki = 831.76 nM T29500 CWT85U 22493254 EC50 < 5011.87 nM T29500 CK8GD3 22493257 EC50 = 316.23 nM T29500 C09UWJ 22493258 EC50 = 5.012 nM T29500 C6BTO5 22493263 EC50 = 63.1 nM T29500 C7NGV2 22493265 EC50 = 316.23 nM T29500 CJ1G5C 22493269 IC50 = 323.59 nM T29500 CR63XU 22493272 EC50 < 5011.87 nM T29500 CGI40S 22493274 EC50 < 5011.87 nM T29500 C3JW1Q 22493280 EC50 = 3.715 nM T29500 CG28DA 22493287 EC50 < 100000 nM T29500 CYHG72 22493289 EC50 = 77.62 nM T29500 CMS13N 22493316 EC50 < 100000 nM T29500 C6ADV8 22493318 EC50 = 6.31 nM T29500 CS4EI0 22493320 EC50 = 79.43 nM T29500 CSF43L 22493325 EC50 < 5011.87 nM T29500 C1QOL5 22493343 EC50 = 39.81 nM T29500 CKIJ24 22493344 EC50 < 100000 nM T29500 C7FCZ5 22493347 EC50 < 5011.87 nM T29500 CDE4R9 22493349 EC50 = 95.5 nM T29500 CSCP16 22493352 EC50 = 1.622 nM T29500 C3N9RK 22493356 EC50 < 100000 nM T29500 C7XEF1 22493359 EC50 = 676.08 nM T29500 C5ZNB0 22493365 EC50 = 79.43 nM T29500 CI1GH6 22493367 EC50 = 199.53 nM T29500 C86PSG 22493372 EC50 < 5011.87 nM T29500 CI42EA 22493379 EC50 = 125.89 nM T29500 CY80ON 22493381 EC50 < 100000 nM T29500 C4LJO9 22493387 EC50 < 100000 nM T29500 CP34UB 22493392 EC50 = 30.2 nM T29500 C9DS1F 22493401 EC50 < 5011.87 nM T29500 CAFG09 22493408 EC50 < 5011.87 nM T29500 C9T5VN 22493411 EC50 < 5011.87 nM T29500 CM86HE 22493415 EC50 < 5011.87 nM T29500 C0NI3J 23290944 Ki = 1051 nM T29500 CL1YH7 23582308 Ki = 251.19 nM T29500 CRN13C 24748804 Ki < 1584.89 nM T29500 C96KDH 24748992 Ki < 1584.89 nM T29500 CH8N1W 24748993 Ki < 794.33 nM T29500 CRGJ52 24749183 Ki < 2511.89 nM T29500 C13GRZ 24749184 Ki < 1995.26 nM T29500 C8ZE6H 24749185 Ki < 3162.28 nM T29500 CWTB59 24749606 Ki < 2511.89 nM T29500 CT93NP 24749721 Ki < 2511.89 nM T29500 CI6W7D 24749841 Ki < 1584.89 nM T29500 C20QND 24749960 Ki < 2511.89 nM T29500 CSXA65 24749962 Ki < 794.33 nM T29500 CUX7C3 24803316 Ki = 316.23 nM T29500 C1QTN4 24803480 Ki > 1995.26 nM T29500 CTU67D 24803482 Ki = 39.81 nM T29500 C31QHW 24803483 Ki = 50.12 nM T29500 C3RYC2 24803638 Ki = 50.12 nM T29500 CI4EA6 24803639 Ki = 125.89 nM T29500 CJ07ES 24803641 Ki = 125.89 nM T29500 C04KHJ 24803797 Ki = 31.62 nM T29500 CY26TH 24803798 Ki = 79.43 nM T29500 C50BOH 24803799 Ki = 100 nM T29500 C2AKX9 24804150 Ki = 39.81 nM T29500 CDC91N 24839550 Ki = 1258.93 nM T29500 C3HK0J 24865725 Ki = 199.53 nM T29500 C0O6FX 24865727 Ki = 158.49 nM T29500 CX6R0P 24894141 Ki = 194.98 nM T29500 C5QG6V 24894147 Ki = 1.413 nM T29500 CW2FG9 24897950 Ki = 5.495 nM T29500 C1VRJ3 25014630 IC50 = 1800 nM T29500 CJOY17 25066019 EC50 > 10000 nM T29500 CF7P2A 25130875 Ki = 281.84 nM T29500 C7P1QS 25130876 Ki = 263.03 nM T29500 C6G5BO 25130877 Ki > 1000 nM T29500 CL8GD3 25130878 Ki > 1000 nM T29500 CT78MG 25130879 Ki = 269.15 nM T29500 C7WXA2 25131192 Ki > 1000 nM T29500 C3UVA0 25131193 Ki = 323.59 nM T29500 C0GM3L 25131196 Ki > 1000 nM T29500 CFUT35 25131198 Ki = 120.23 nM T29500 C1Y3TS 25131871 Ki > 1000 nM T29500 CFJ6Y9 25131876 Ki = 56.23 nM T29500 CNQX42 25132217 Ki > 1000 nM T29500 C7WE4Y 25132564 Ki > 1000 nM T29500 C6K1TB 25132565 Ki > 1000 nM T29500 CJ19KC 25132566 Ki = 302 nM T29500 CNO83H 25181488 Ki = 21.88 nM T29500 CEYF08 25181489 Ki = 52.48 nM T29500 CAM63X 42618195 IC50 > 1000 nM T29500 C8K4UF 42618197 IC50 > 1000 nM T29500 CJ3NP5 42636941 IC50 = 144.54 nM T29500 CW2DP3 44123711 Ki = 125.89 nM T29500 C2HPM1 44213730 Ki = 158.49 nM T29500 C2DS9L 44213782 Ki = 940 nM T29500 CTR42S 44219718 EC50 > 10000 nM T29500 CB2HY8 44219719 EC50 > 10000 nM T29500 C4T7ZI 44222842 Ki = 22.39 nM T29500 C9ROX7 44267817 Ki = 10000 nM T29500 C0L4TU 44267884 Ki = 2244 nM T29500 CF2DH7 44267890 Ki = 10000 nM T29500 CEL7U6 44267912 Ki = 10000 nM T29500 CF51JW 44268966 Ki = 15.8 nM T29500 C89FEL 44269124 EC50 < 100000 nM T29500 CVE83T 44271661 EC50 = 0.3981 nM T29500 C7P2AH 44271931 EC50 < 100000 nM T29500 CSQ5L6 44271932 EC50 = 39.81 nM T29500 C5UA4W 44273916 Ki = 15 nM T29500 CMH52E 44275255 Ki = 281.84 nM T29500 C7Q2JD 44275526 Ki = 173.78 nM T29500 CPK7B3 44284333 Ki = 20.42 nM T29500 CZPD80 44288485 Ki = 170 nM T29500 C5UIM4 44288492 Ki > 3000 nM T29500 CL3RI0 44288729 Ki > 2000 nM T29500 CTR4Z6 44288740 Ki = 840 nM T29500 C4K6RC 44288741 Ki > 3000 nM T29500 CQP9B7 44288754 Ki = 1700 nM T29500 CZ5P6U 44288769 Ki = 842 nM T29500 CV8G1J 44288792 Ki = 870 nM T29500 CQ40MA 44288794 Ki = 2000 nM T29500 CX7BT8 44288810 Ki = 570 nM T29500 CA16JS 44288815 Ki = 650 nM T29500 C4KND2 44288816 Ki = 1100 nM T29500 CT7IB6 44288841 Ki = 34 nM T29500 CEM2T4 44288843 Ki > 2000 nM T29500 CZ7O4D 44288847 Ki > 2000 nM T29500 C8EJ9B 44288857 Ki = 3300 nM T29500 CKA01M 44288858 Ki > 2000 nM T29500 CL4X9R 44288864 Ki > 2000 nM T29500 C6DYQ1 44288874 Ki = 805 nM T29500 CAG7E1 44288877 Ki > 2000 nM T29500 CQ74LV 44288917 Ki = 1040 nM T29500 CQ3Y5R 44288945 Ki = 37 nM T29500 CZDR39 44288995 Ki = 960 nM T29500 C92FEY 44289026 Ki = 1900 nM T29500 C9HMK3 44289034 Ki = 680 nM T29500 C5ZL4A 44289035 Ki = 425 nM T29500 C71XMR 44289047 Ki = 670 nM T29500 CW5C4G 44289058 Ki = 1200 nM T29500 C62NWB 44289089 Ki = 910 nM T29500 C37GEA 44289100 Ki = 54 nM T29500 C1ES5Y 44289103 Ki = 1200 nM T29500 CZS9B7 44289107 Ki = 330 nM T29500 CZSM05 44289112 Ki = 570 nM T29500 C51NLQ 44289248 Ki = 1.148 nM T29500 CWC49F 44289261 Ki = 12.3 nM T29500 C14WMG 44289321 Ki = 6.6 nM T29500 CQW1Z3 44289344 Ki = 23 nM T29500 CFO29U 44289346 Ki > 2000 nM T29500 C1JX5M 44289437 Ki = 1.23 nM T29500 CIM92E 44289525 Ki = 51.38 nM T29500 CF1UW9 44294569 Ki = 22.1 nM T29500 CBS42M 44294957 Ki = 210 nM T29500 CW6D7V 44294958 Ki = 350 nM T29500 CMQ6G5 44295044 Ki = 970 nM T29500 C9XAB7 44295046 Ki = 130 nM T29500 C9MQ4B 44295133 Ki = 120 nM T29500 CNQ82T 44295170 Ki = 1200 nM T29500 C9Y3GE 44295192 Ki = 300 nM T29500 C4KB8E 44295193 Ki = 390 nM T29500 C9UW2H 44295218 Ki = 340 nM T29500 CWJ13T 44298447 Ki = 15.85 nM T29500 C0F8LH 44298611 Ki = 15.85 nM T29500 C0M5BZ 44298624 Ki = 10 nM T29500 C17AXP 44298626 Ki = 39.81 nM T29500 CA19EZ 44298644 Ki = 398.11 nM T29500 C0QLW1 44298650 Ki = 100 nM T29500 CO6K1V 44298664 Ki = 5.012 nM T29500 CMI12L 44298671 Ki = 158.49 nM T29500 CBJ31S 44298694 Ki = 100 nM T29500 CUO47C 44298734 Ki = 158.49 nM T29500 CDLJ86 44298735 Ki = 100 nM T29500 C4N1EM 44298746 Ki = 63.1 nM T29500 C1V0RE 44298747 Ki = 6.31 nM T29500 C1H2MT 44298762 Ki = 199.53 nM T29500 C3X6RY 44298770 Ki = 50.12 nM T29500 C9TR2K 44298780 Ki = 251.19 nM T29500 CX90HD 44299835 Ki = 290 nM T29500 C6HO4W 44299945 Ki = 120 nM T29500 CG82KA 44299973 Ki = 14 nM T29500 CL62DY 44299974 Ki = 51 nM T29500 C0LF1S 44299975 Ki = 28 nM T29500 CM8KV2 44300018 Ki = 86.96 nM T29500 CY8J6F 44300087 Ki = 91 nM T29500 CYV46S 44300107 Ki = 70 nM T29500 CLHT17 44300111 Ki = 1300 nM T29500 C2WP7S 44300129 Ki = 350 nM T29500 CH59JV 44300159 Ki = 730 nM T29500 C8K3AP 44300165 Ki = 130 nM T29500 CSA23P 44300166 Ki = 130 nM T29500 C3YDV9 44300170 Ki = 36 nM T29500 CW56GZ 44301572 Ki > 2000 nM T29500 CH34AY 44301573 Ki = 1500 nM T29500 CIPQ70 44301680 Ki > 2000 nM T29500 C5EZ6B 44301681 Ki = 1800 nM T29500 C6R2DV 44308443 Ki > 5000 nM T29500 C8M4HW 44308466 Ki = 592 nM T29500 CPUO39 44308654 Ki = 2569 nM T29500 C6G8ZC 44311789 Ki = 104712.85 nM T29500 C5L1WN 44312036 Ki < 100000 nM T29500 CT46CK 44312037 Ki = 60255.96 nM T29500 C3XFH4 44312198 Ki = 141253.75 nM T29500 C3BQW5 44312563 Ki = 1.58 nM T29500 CKU7Y6 44316072 Ki = 2770 nM T29500 CG2UB8 44316098 Ki = 3080 nM T29500 C2PR8V 44318000 Ki > 5000 nM T29500 CZ5M4K 44318075 Ki > 5000 nM T29500 C8JKO2 44318081 Ki = 1400 nM T29500 C3J9XH 44324405 Ki = 7.9 nM T29500 CT7DN4 44327688 Ki < 10000 nM T29500 CGP40I 44329083 EC50 < 5011.87 nM T29500 CES26R 44329133 EC50 = 12.59 nM T29500 CR3N5S 44329318 EC50 < 5011.87 nM T29500 CZ21VE 44329481 EC50 < 5011.87 nM T29500 C4ZV9T 44329701 EC50 = 79.43 nM T29500 CBZ84S 44329703 EC50 = 63.1 nM T29500 CQY03V 44329738 EC50 < 5011.87 nM T29500 C7Z2HM 44329739 EC50 < 5011.87 nM T29500 CS2WN0 44329788 EC50 < 5011.87 nM T29500 C5AG1U 44329790 EC50 = 158.49 nM T29500 C14RBX 44329796 EC50 = 25.12 nM T29500 CG60QK 44329797 EC50 < 5011.87 nM T29500 CIJ52V 44329992 Ki < 10000 nM T29500 C4Q3HY 44329993 Ki = 7762.47 nM T29500 C6US9E 44330880 Ki = 137 nM T29500 C2N0GV 44331079 Ki = 53 nM T29500 C02JUQ 44331090 Ki = 149 nM T29500 CU2H1F 44331136 Ki = 24 nM T29500 C5SLE2 44331150 Ki = 53 nM T29500 CK5R0A 44331169 Ki = 175 nM T29500 CGJB37 44331174 Ki = 49 nM T29500 CI9UV3 44331198 Ki = 55 nM T29500 C4RJ7I 44331277 Ki = 48 nM T29500 CP9B2K 44340834 Ki = 309.03 nM T29500 CB23YQ 44340835 Ki = 93.33 nM T29500 CC25ZK 44340836 Ki = 30.2 nM T29500 CZBQ72 44340850 Ki = 19.05 nM T29500 CTM65V 44340854 Ki = 43.65 nM T29500 CQ3WH6 44341114 Ki = 89.13 nM T29500 CO5T9G 44343173 EC50 < 5011.87 nM T29500 C0DS6V 44343235 EC50 < 100000 nM T29500 CK1QJ5 44343236 EC50 = 100 nM T29500 CV5N1T 44343243 EC50 < 5011.87 nM T29500 C84GDJ 44343244 EC50 < 5011.87 nM T29500 CV8LE9 44343245 EC50 < 5011.87 nM T29500 CX8J0Y 44343247 EC50 = 316.23 nM T29500 C71WZX 44343251 EC50 < 100000 nM T29500 C19JFN 44343257 EC50 < 100000 nM T29500 C17HRU 44343275 EC50 < 5011.87 nM T29500 C6ZU5G 44343410 EC50 = 25.12 nM T29500 CQR12J 44343520 EC50 < 5011.87 nM T29500 CFQ32B 44343524 IC50 < 30199.52 nM T29500 CZ2X3A 44352155 EC50 < 100000 nM T29500 C3I9DE 44358574 Ki = 26.4 nM T29500 C2WYI7 44361064 Ki = 18.62 nM T29500 C8OM7A 44362013 EC50 < 100000 nM T29500 CK6S1Y 44362145 EC50 < 100000 nM T29500 C7FHB4 44362146 EC50 = 15.85 nM T29500 CSFJ14 44362149 EC50 = 12.59 nM T29500 CEZ8K0 44362150 EC50 = 79.43 nM T29500 CK8U9S 44362185 EC50 = 79.43 nM T29500 CHL40X 44362194 EC50 = 5.012 nM T29500 C3CF8S 44362195 EC50 = 1 nM T29500 C78CEY 44362196 EC50 = 19.95 nM T29500 C3AU6V 44362208 EC50 = 3.981 nM T29500 CH9B3A 44362286 EC50 = 10 nM T29500 CF6H7S 44362287 EC50 < 100000 nM T29500 CI6DH4 44362288 EC50 = 630.96 nM T29500 C2SBP1 44362289 EC50 < 100000 nM T29500 CH79ZL 44362510 EC50 < 100000 nM T29500 C0GR4S 44362511 EC50 < 100000 nM T29500 C1U0TR 44362523 EC50 < 100000 nM T29500 CEQD62 44362541 EC50 < 100000 nM T29500 CU0E7G 44362633 Ki = 1450 nM T29500 C94ORM 44362867 Ki = 860 nM T29500 CZ1KQ9 44369351 EC50 = 5.754 nM T29500 C1Y7OL 44369431 EC50 = 112.2 nM T29500 C03STZ 44369434 EC50 = 46.77 nM T29500 C6W2MT 44369646 EC50 < 100000 nM T29500 CDR8C3 44369647 EC50 < 100000 nM T29500 C4B0OI 44397588 Ki = 199.53 nM T29500 C5FP0R 44397589 Ki = 316.23 nM T29500 CE3G8U 44397670 Ki = 316.23 nM T29500 C27FZA 44417706 Ki = 891.25 nM T29500 C31WOV 44417713 Ki = 85.11 nM T29500 C85GUJ 44420408 Ki = 10.72 nM T29500 CHIA46 44420412 Ki = 91.2 nM T29500 C6I3MN 44420418 Ki = 19054.61 nM T29500 CQV5N7 44420419 Ki = 602.56 nM T29500 CSQ5H2 44420423 Ki = 83.18 nM T29500 C1CFB6 44420428 Ki = 17.38 nM T29500 CAW15U 44420431 Ki = 17.38 nM T29500 C7C4QE 44426404 Ki = 275 nM T29500 CE3XQ2 44426405 Ki = 76 nM T29500 C21KYB 44428845 Ki = 0.309 nM T29500 C91BHJ 44428846 Ki = 0.871 nM T29500 CCLI02 44428847 Ki = 1.38 nM T29500 CE08JS 44428848 Ki = 0.2399 nM T29500 CVH1Z5 44428849 Ki = 3.162 nM T29500 CY26IH 44428850 Ki = 5.888 nM T29500 CRN18J 44428851 Ki = 0.4898 nM T29500 CBK87I 44431173 Ki = 4108 nM T29500 CX3D0B 44431174 Ki = 1082 nM T29500 C9HD0G 44431180 Ki = 15 nM T29500 CB3A8T 44431184 Ki = 46.5 nM T29500 C09VIB 44431192 Ki = 44.6 nM T29500 C43SCL 44431194 Ki = 22.4 nM T29500 C4G7QF 44431545 Ki = 111 nM T29500 C8OP5V 44431546 Ki = 31 nM T29500 C0B5TC 44431547 Ki = 103 nM T29500 CCXB24 44431548 Ki = 201 nM T29500 C5QI0V 44431551 Ki = 108 nM T29500 C2R4TP 44431553 Ki = 222 nM T29500 COIS42 44431554 Ki = 150 nM T29500 C0APQ4 44431555 Ki = 195 nM T29500 CJT34W 44431557 Ki = 174 nM T29500 CF76RP 44431560 Ki = 106 nM T29500 CY8C0V 44431562 Ki = 153 nM T29500 C2UD6M 44431564 Ki = 162 nM T29500 C4J0TG 44431574 Ki = 162 nM T29500 C0C8TU 44431587 Ki = 42 nM T29500 C1QV6S 44431590 Ki = 258 nM T29500 CF3ST7 44431594 Ki = 85 nM T29500 CA9O2E 44431599 Ki = 167 nM T29500 CX9YA2 44431602 Ki = 177 nM T29500 C9OSE8 44431607 Ki = 120 nM T29500 CT0LP1 44431611 Ki = 101 nM T29500 C46NHX 44431612 Ki = 1855 nM T29500 C3IA4W 44431613 Ki = 364 nM T29500 C5QJ8S 44431614 Ki = 601 nM T29500 CXD1Q9 44431615 Ki = 952 nM T29500 C0WPS6 44431616 Ki = 82 nM T29500 C4SZA3 44431617 Ki = 192 nM T29500 CE6L0D 44431618 Ki = 169 nM T29500 CS9N3Q 44431620 Ki = 125 nM T29500 CEWQ41 44433348 Ki = 109 nM T29500 C64POV 44449245 EC50 = 600 nM T29500 CX7Z6I 44449247 EC50 > 10000 nM T29500 CO9NC7 44449248 EC50 > 10000 nM T29500 C1P3XZ 44449249 EC50 > 10000 nM T29500 CN9BI4 44449276 EC50 > 10000 nM T29500 CYM30S 44449277 EC50 > 10000 nM T29500 CS5WB3 44449278 EC50 > 10000 nM T29500 CH74NV 44449303 EC50 > 10000 nM T29500 C8VO6A 44449304 EC50 > 10000 nM T29500 CI4T2K 44449305 EC50 > 10000 nM T29500 C70SEG 44449306 EC50 > 10000 nM T29500 C0M7UN 44449337 EC50 > 10000 nM T29500 C4THN7 44449338 EC50 > 10000 nM T29500 C1O6QI 44449657 EC50 > 10000 nM T29500 C6QCN8 44449686 EC50 > 10000 nM T29500 CH5RL7 44449690 EC50 > 10000 nM T29500 CS3LB0 44449691 EC50 > 10000 nM T29500 CFL25O 44449692 EC50 > 10000 nM T29500 CSZB25 44449694 EC50 > 10000 nM T29500 CJ8WL7 44449723 EC50 > 10000 nM T29500 C8XHB5 44449724 EC50 > 10000 nM T29500 C6ZG3O 44449725 EC50 = 902 nM T29500 CMLE59 44449730 EC50 > 10000 nM T29500 CZL97F 44455426 Ki = 325 nM T29500 C12XGE 44456400 Ki > 10000 nM T29500 CGO23X 44460394 Ki > 5000 nM T29500 CLVD72 44460423 Ki = 2205 nM T29500 C7T2KE 44460449 Ki > 5000 nM T29500 CVJ72X 44460477 Ki > 5000 nM T29500 CT5M7N 44460522 Ki > 5000 nM T29500 CV3IW1 44461012 Ki = 676 nM T29500 C1PI3F 44462130 Ki = 2200 nM T29500 CJ10OZ 44531812 Ki = 323.59 nM T29500 CT85QK 44538690 Ki = 104 nM T29500 CAR23X 44568818 Ki = 141.25 nM T29500 CAO31F 44568917 Ki = 74.13 nM T29500 CE3GV8 44568918 Ki = 125.89 nM T29500 CVF30Y 44574044 EC50 > 10000 nM T29500 CCD72N 44574045 EC50 > 10000 nM T29500 CMS20J 44574074 EC50 > 6500 nM T29500 C92YUA 44574075 EC50 > 1400 nM T29500 C9NU2C 44574076 EC50 > 10000 nM T29500 CX4Y0K 44574078 EC50 = 760 nM T29500 CU9X8G 44574079 EC50 > 10000 nM T29500 CAT57X 44574103 EC50 > 10000 nM T29500 CXZ0J3 44574104 EC50 > 10000 nM T29500 CES4X0 44574105 EC50 > 10000 nM T29500 C62AYR 44574106 EC50 > 10000 nM T29500 CX98MY 44574107 EC50 > 10000 nM T29500 CDER54 44574132 EC50 > 10000 nM T29500 C4S2OQ 44574133 EC50 > 10000 nM T29500 C96NQZ 44574134 EC50 = 990 nM T29500 CKR69S 44574135 EC50 > 10000 nM T29500 C4WZG9 44574136 EC50 > 10000 nM T29500 CL37FD 44574137 EC50 > 10000 nM T29500 CG0RM2 44574138 EC50 > 10000 nM T29500 CD87ZE 44574834 EC50 > 10000 nM T29500 C2YF8O 44574874 EC50 > 10000 nM T29500 CFQJ71 44574875 EC50 > 10000 nM T29500 CB1R3O 44574876 EC50 > 10000 nM T29500 CR8SF7 44574877 EC50 > 10000 nM T29500 CN94EW 44574878 EC50 > 10000 nM T29500 C8L6CN 44574934 EC50 > 10000 nM T29500 CVN8Z4 44574935 EC50 = 1100 nM T29500 C9QAM5 44574936 EC50 > 10000 nM T29500 CV06SB 44574938 EC50 > 10000 nM T29500 C3QWO0 44574986 EC50 = 1770 nM T29500 C4XHI5 44574989 EC50 > 10000 nM T29500 CYAI96 44575544 IC50 = 215 nM T29500 C5NS6H 44581972 Ki = 630.96 nM T29500 CK8Z1P 44581973 Ki = 562.34 nM T29500 C3UQ9Z 44581974 Ki = 1445.44 nM T29500 CRCH48 44582675 Ki = 500 nM T29500 CEJ4R8 44582676 Ki = 550 nM T29500 C5QB4K 44582678 Ki > 10000 nM T29500 C9F6EB 44593557 EC50 > 10000 nM T29500 C51AJZ 44593577 EC50 > 10000 nM T29500 CDA54Q 44593580 EC50 > 10000 nM T29500 C1SN7Y 44593709 Ki = 66.07 nM T29500 CWO70X 45260703 Ki = 794.33 nM T29500 C4VOW6 45260704 EC50 = 61.66 nM T29500 CQ0R5Y 45264581 EC50 = 2.188 nM T29500 C39CDN 45264638 EC50 = 13.8 nM T29500 C0F4TJ 45268939 Ki = 0.4169 nM T29500 CMNA70 45358442 Ki = 158.49 nM T29500 C05PBD 46176231 IC50 > 10000 nM T29500 C0ABR3 46846073 Ki > 1000 nM T29500 C7ZEI6 46881382 Ki = 117.49 nM T29500 CN0Q2A 46881443 Ki = 58.88 nM T29500 CGX02N 46881444 Ki = 41.69 nM T29500 C2MC4K 46881463 Ki = 316.23 nM T29500 CSQ4C9 46881468 Ki = 251.19 nM T29500 C4U6RH 46881493 Ki = 239.88 nM T29500 CV7R9S 46881494 Ki = 100 nM T29500 C24QFO 46882032 Ki > 1000 nM T29500 C3GQW6 46882033 Ki > 1000 nM T29500 CPG6U5 46882034 Ki = 19.95 nM T29500 CYB37P 46882085 Ki = 53.7 nM T29500 CD8CX3 46882086 Ki = 446.68 nM T29500 C57GAO 46882087 Ki = 138.04 nM T29500 CV3QW9 46882088 Ki = 173.78 nM T29500 C5ZDY3 46915370 Ki = 758 nM T29500 CI4XZ1 46934637 Ki = 51.29 nM T29500 CK1Z0M 46934639 Ki = 128.82 nM T29500 CU0TB9 46934641 Ki = 18.2 nM T29500 CR6JV7 46934643 Ki = 72.44 nM T29500 C14ZLO 46934645 Ki = 223.87 nM T29500 C2N9JZ 46934787 Ki = 85.11 nM T29500 CI4U0L 46934789 Ki = 131.83 nM T29500 C8HVG6 46934791 Ki = 46.77 nM T29500 CA51JI 46934793 Ki = 10 nM T29500 CB4Z7D 46934945 Ki = 9.333 nM T29500 CV93BN 46945445 Ki > 10000 nM T29500 C8VUO2 49781004 Ki = 912.01 nM T29500 C0LAT9 49781005 Ki = 63.1 nM T29500 C12UVE 49781006 Ki = 39.81 nM T29500 CW1V4K 49781007 Ki = 11.48 nM T29500 CF9L7Z 49781008 Ki = 316.23 nM T29500 CQ2EN5 49781222 Ki = 6.166 nM T29500 CV62OU 49781223 Ki = 40.74 nM T29500 C3I5HP 49781224 Ki = 8.913 nM T29500 CF5CO4 49781228 Ki = 1.047 nM T29500 CW5X6A 49781887 Ki = 14.79 nM T29500 C2LZJ0 49783209 Ki > 10000 nM T29500 C57SMG 49783415 Ki = 4228 nM T29500 C0TG6I 49783419 Ki = 9076 nM T29500 C0D5GI 49796077 Ki = 257.04 nM T29500 C6ZRD7 49797187 Ki = 426.58 nM T29500 C63FGJ 49797190 Ki = 398.11 nM T29500 C6IW4Q 49862238 Ki > 1000 nM T29500 CZ2SA8 49864841 Ki = 3.162 nM T29500 C2RY0J 50878551 Ki < 10000 nM T29500 C1W6TV 50898777 Ki > 10000 nM T29500 CXMZ73 50898778 Ki > 10000 nM T29500 C8EU7J 50905381 Ki = 1.905 nM T29500 CW7FI3 50905585 Ki = 2.089 nM T29500 CIL56G 50905588 Ki = 67.61 nM T29500 C5M6VO 50905589 Ki = 31.62 nM T29500 CX48AD 51002362 Ki = 3791 nM T29500 CE4KP1 51050257 Ki > 10000 nM T29500 CQG7X2 51349173 EC50 > 10000 nM T29500 CF9V1U 52937018 Ki = 316.23 nM T29500 CS3BJ7 52937119 Ki = 79.43 nM T29500 C93QXP 52937222 Ki = 6.31 nM T29500 CPF7V0 52937223 Ki = 316.23 nM T29500 CYG24L 52937526 Ki = 158.49 nM T29500 CL8QZ3 52937527 Ki = 398.11 nM T29500 CM36PE 52937629 Ki > 1995.26 nM T29500 CRV61I 52937630 Ki = 79.43 nM T29500 CEKB47 52937631 Ki = 15.85 nM T29500 CZ0C5B 52937632 Ki > 1995.26 nM T29500 CVX7U2 52937633 Ki > 1995.26 nM T29500 C3ZX1Q 52937634 Ki > 1995.26 nM T29500 CY4N8T 52937728 Ki = 398.11 nM T29500 C83WTP 52937729 Ki = 630.96 nM T29500 CQDS92 52937730 Ki > 1995.26 nM T29500 CR0KW9 52937731 Ki = 501.19 nM T29500 C2UV5S 52937732 Ki = 316.23 nM T29500 C6XHP8 52937733 Ki > 1995.26 nM T29500 C3B5HN 52937734 Ki > 1995.26 nM T29500 CK52QG 52937828 Ki = 199.53 nM T29500 CFV4D0 52937829 Ki = 1000 nM T29500 C9MBQ2 52937830 Ki = 19.95 nM T29500 CLW3B0 52940951 Ki = 7.943 nM T29500 CWYS78 52941004 Ki = 12.59 nM T29500 CE0X9W 52941056 Ki = 100 nM T29500 CR8MI3 52941512 Ki = 33.11 nM T29500 C40WVE 52941624 Ki = 19.95 nM T29500 CV7HZ6 52942047 Ki = 173.78 nM T29500 C5Y3VS 52942152 Ki = 5.012 nM T29500 CO9J6M 52943356 Ki = 5.012 nM T29500 CH3YE5 52943739 Ki = 39.81 nM T29500 C70LBS 52944548 Ki = 16.6 nM T29500 CRL3P0 52944615 Ki = 79.43 nM T29500 C4N6ET 52944674 Ki = 100 nM T29500 CDQ27E 52945156 Ki = 15.85 nM T29500 CPI9F4 52945803 Ki = 0.7943 nM T29500 CGZ1R7 52947088 Ki = 100 nM T29500 CNH57S 52947579 Ki = 0.5012 nM T29500 CX04NC 52948119 Ki = 70.79 nM T29500 C9YBJ3 52948823 Ki = 6.918 nM T29500 C7WN4S 52948958 Ki = 3.548 nM T29500 CCQZ15 52949448 Ki = 6.761 nM T29500 C5W7SH 52950140 Ki = 177.83 nM T29500 CGY45S 53248361 Ki = 185 nM T29500 CE9L8G 53248365 Ki = 25 nM T29500 C4H5JI 53327748 Ki = 3.981 nM T29500 C1YX4A 53327991 Ki = 7.943 nM T29500 CUP50Y 53327992 Ki = 19.95 nM T29500 CZ1B6D 53328115 Ki = 7413.1 nM T29500 CT0D9O 53328116 Ki = 2238.72 nM T29500 CGB3U6 53328311 Ki = 112.2 nM T29500 CIWJ61 53328312 Ki = 112.2 nM T29500 CW36HN 53328313 Ki = 331.13 nM T29500 C6NUW4 53328314 Ki = 30.2 nM T29500 C7XCQ4 53328315 Ki = 107.15 nM T29500 CJ7TY9 53328316 Ki = 97.72 nM T29500 C76NJW 53328503 Ki = 112.2 nM T29500 CB1D8L 53328504 Ki = 10000 nM T29500 CY9JI7 53328505 Ki = 125.89 nM T29500 C5FHA1 53328506 Ki = 134.9 nM T29500 CCM7S9 53328507 Ki = 245.47 nM T29500 C7YN2M 53328508 Ki = 128.82 nM T29500 CD7EB0 53328684 Ki = 208.93 nM T29500 CQGE30 53328685 Ki = 128.82 nM T29500 CNSU94 53328686 Ki = 194.98 nM T29500 CY51RC 53328687 Ki = 151.36 nM T29500 C9L0ZI 53328872 Ki = 5011.87 nM T29500 C67YNQ 53328873 Ki = 234.42 nM T29500 CMOZ61 53475319 Ki = 666 nM T29500 CGX1W2 53779053 Ki = 74 nM T29500 C6W1RA 56649648 Ki = 176 nM T29500 C2SW7J 56649649 Ki = 110 nM T29500 CQTR49 56649650 Ki = 38 nM T29500 CA6B2I 56668277 Ki = 1900 nM T29500 CCW38Z 56945164 Ki = 74.13 nM T29500 CN6XE8 56945165 Ki = 165.96 nM T29500 CPE6C7 56945166 Ki = 288.4 nM T29500 C4L7GW 56945167 Ki = 245.47 nM T29500 CL68PZ 56946472 Ki = 123.03 nM T29500 CJ98DO 56946474 Ki = 39.81 nM T29500 CB8J2F 56946573 Ki = 8.913 nM T29500 CCBY53 56946575 Ki > 1000 nM T29500 CMO0U3 56946577 Ki > 1000 nM T29500 CJZ3P4 56946579 Ki = 141.25 nM T29500 CXUW26 56961460 IC50 < 5 nM T29500 CX74AS 56961506 IC50 < 5 nM T29500 C9WP3O 56961507 Ki = 7.3 nM T29500 C1TC7Q 56963799 Ki > 10000 nM T29500 CDTG05 57393527 Ki = 6.761 nM T29500 C8EFT7 57402251 Ki > 1000 nM T29500 CT89JH 57780007 Ki > 1995.26 nM T29500 CT8RO7 57780008 Ki = 15.85 nM T29500 C5RIN4 57780016 Ki = 79.43 nM T29500 CE9WC0 57780017 Ki = 199.53 nM T29500 C1W4SB 57780018 Ki > 1995.26 nM T29500 CT96WD 57780020 Ki = 398.11 nM T29500 C3XL7O 66561967 Ki > 10000 nM T29500 C1SBP9 69781970 Ki = 0.3802 nM T29500 CCD2L1 69782867 Ki = 0.1514 nM T29500 CBQ8P4 71449250 Ki = 125.89 nM T29500 C6SN2P 71449516 Ki = 398.11 nM T29500 C9VZ8J 71450550 Ki = 3490 nM T29500 CFS69A 71450901 Ki = 12.59 nM T29500 CB83YL 71451044 Ki = 100 nM T29500 C75EQJ 71452768 Ki = 48 nM T29500 C0YXD3 71452871 Ki = 10 nM T29500 CY7NM9 71452872 Ki = 158.49 nM T29500 C9O1YZ 71454559 Ki = 1.63 nM T29500 C4JN5I 71454639 Ki = 19.95 nM T29500 C31VFN 71454865 Ki = 30.9 nM T29500 C8YH0J 71455083 Ki = 296 nM T29500 C6G2HC 71455894 Ki = 2766 nM T29500 CMBU21 71456359 Ki = 12.59 nM T29500 CVT39B 71456360 Ki = 316.23 nM T29500 CK87DI 71456361 Ki = 251.19 nM T29500 C7MNB5 71457264 Ki = 955.4 nM T29500 CP7JI0 71457691 Ki = 536 nM T29500 C3VMS0 71458203 Ki = 25.12 nM T29500 C8T5EJ 71458204 Ki = 50.12 nM T29500 CZ6BX7 71458205 Ki = 39.81 nM T29500 CORB94 71458492 Ki = 33.88 nM T29500 CK5T4P 71459604 Ki > 10000 nM T29500 CEBC62 71461781 Ki = 15.85 nM T29500 C9DJ1V 71461782 Ki = 7.943 nM T29500 CA6NI7 71462043 Ki = 2.188 nM T29500 CD9G8B 71521478 Ki = 1659.59 nM T29500 CSV0G5 71521479 Ki = 416.87 nM T29500 CGN2M7 71521480 Ki = 169.82 nM T29500 CDS15J 71659980 Ki = 5.37 nM T29500 CH6J4G 71817545 Ki = 489.78 nM T29500 CH54DW 71817546 Ki = 21.88 nM T29500 C3NO8R 71817548 Ki = 35.48 nM T29500 CRTD80 71817857 Ki = 1905.46 nM T29500 CBTX18 71817858 Ki = 162.18 nM T29500 CRYP87 71817860 Ki = 371.54 nM T29500 CC65OA 73213195 Ki > 10000 nM T29500 CW83DK 73213196 Ki = 2238.72 nM T29500 CCV91B 73346042 Ki = 26.8 nM T29500 CY60RD 73347826 Ki = 3442 nM T29500 CX01MD 73349178 Ki = 125.89 nM T29500 CM63WH 73352416 Ki = 9.4 nM T29500 CAI63V 73355417 Ki = 6196 nM T29500 CBW1D8 73356785 Ki = 28.84 nM T29500 C2E7QW 75201901 Ki = 9200 nM T29500 C8IDL3 75306277 Ki > 1000 nM T29500 CFN6P8 76071738 IC50 > 10000 nM T29500 CW61JI 76071739 IC50 > 10000 nM T29500 C04HNK 76308473 Ki = 0.871 nM T29500 C8M3OX 76323009 Ki = 0.871 nM T29500 COT51G 76326561 Ki = 1.38 nM T29500 CFV87U 76330228 Ki = 0.309 nM T29500 C3Z1TP 78815633 Ki = 10.23 nM T29500 CL9AI7 85469698 IC50 = 875.3 nM T29500 CGO74F 85469753 IC50 = 1003 nM T29500 C91LTS 85469754 IC50 = 199 nM T29500 CS9DG8 85469755 IC50 = 787.5 nM T29500 CU6R1L 85469756 IC50 = 406.2 nM T29500 CTRN10 85469757 IC50 = 34.76 nM T29500 CU3P0H 85469808 IC50 = 1007 nM T29500 C74PRV 85469809 IC50 = 121.9 nM T29500 CUOH37 85469811 IC50 = 781.5 nM T29500 CKNG20 85469812 IC50 = 433.3 nM T29500 C6-MAR-04 85469868 IC50 = 769.4 nM T29500 CJQ9O7 85469869 IC50 = 12.57 nM T29500 C4HA3I 85469870 IC50 = 948.8 nM T29500 C9NL2S 85469871 IC50 = 1876 nM T29500 C1J0GW 85469872 IC50 = 794.4 nM T29500 CVM3B2 85469873 IC50 = 250.4 nM T29500 CYI5J6 85469930 IC50 = 31.62 nM T29500 CZI3Y2 85469931 IC50 = 19.69 nM T29500 CAS6Y8 85469932 IC50 = 100.9 nM T29500 C7PXK3 85469933 IC50 = 28.91 nM T29500 C7XI0F 85469934 IC50 = 684 nM T29500 CLBA19 86344174 IC50 = 2862 nM T29500 CL9GY7 90645592 Ki = 10 nM T29500 CI49HV 90645593 Ki = 28.18 nM T29500 C41AGZ 90645594 Ki = 33.88 nM T29500 C1L0PW 90645595 Ki = 36.31 nM T29500 C7JL5G 90645596 Ki = 2.692 nM T29500 C89TJI 90645597 Ki = 0.8318 nM T29500 CHBC38 90645598 Ki = 1.905 nM T29500 C4MLA7 90645599 Ki = 6.457 nM T29500 C0WXR7 90645600 Ki = 7.413 nM T29500 CN8TF6 90645601 Ki = 1.66 nM T29500 CKN56Z 90645602 Ki = 38.9 nM T29500 CYQ3M8 90645603 Ki = 30.2 nM T29500 C45MSD 90645604 Ki = 19.05 nM T29500 C4I6EW 90645605 Ki = 6.457 nM T29500 CH92LD 90645606 Ki = 7.586 nM T29500 C7YQM3 101333429 Ki = 234 nM T29500 CE0ZC6 101876962 Ki = 39.81 nM T29500 CJ15CM 102012413 Ki = 76 nM T29500 CA43MY 117839022 IC50 = 1736 nM T29500 CI7NQ9 118716698 Ki = 141.25 nM T29500 CGO9W4 118716699 Ki = 323.59 nM T29500 CVDI36 118716700 Ki = 16.6 nM T29500 C94AFL 118716701 Ki = 478.63 nM T29500 CTX92K 118716702 Ki = 288.4 nM T29500 CG02WP 118716703 Ki = 42.66 nM T29500 CTNL85 118716704 Ki = 154.88 nM T29500 CM1Y8W 118716705 Ki = 1000 nM T29500 C42MOT 118716706 Ki = 67.61 nM T29500 C78ARU 118716707 Ki = 63.1 nM T29500 CO5TG3 118716708 Ki = 158.49 nM T29500 CNF78L 118716709 Ki = 109.65 nM T29500 C9CB1Q 118716710 Ki = 158.49 nM T29500 C3F6EQ 118716711 Ki = 1000 nM T29500 C0L6YO 118716712 Ki = 1000 nM T29500 CX2AC4 118716713 Ki = 85.11 nM T29500 CL1EU8 118716714 Ki = 8.318 nM T29500 C0V7GJ 118716715 Ki = 69.18 nM T29500 CRBI65 118716716 Ki = 147.91 nM T29500 C70IPZ 118716717 Ki = 109.65 nM T29500 CBI30N 118716718 Ki = 69.18 nM T29500 C7UBN8 118716719 Ki = 85.11 nM T29500 CV8HA2 118716720 Ki = 363.08 nM T29500 C30ZJB 118716721 Ki = 81.28 nM T29500 C58MND 118716722 Ki = 239.88 nM T29500 CO6T4G 118716723 Ki = 128.82 nM T29500 C8RVX4 118717455 Ki = 19 nM T29500 C5IM1N 118717456 Ki = 47.86 nM T29500 CBCU90 118717457 Ki = 50 nM T29500 CN4LJ2 118717458 Ki = 151 nM T29500 CZ35PU 118717459 Ki = 147.91 nM T29500 C9BP7A 118717460 Ki = 51 nM T29500 CFCM61 118717461 Ki = 34.67 nM T29500 C8C6ZW 118717462 Ki = 154.88 nM T29500 CR8Z0F 118718431 Ki > 2000 nM T29500 CON3I0 118727908 EC50 = 3.5 nM T29500 C8Z0PK 118727909 EC50 = 131.1 nM T29500 CQL0Y3 118727912 EC50 = 165.3 nM T29500 C97AZR 118727914 EC50 = 46.9 nM T29500 CT4CW7 118727915 EC50 = 2.53 nM T29500 C0WSD7 118727918 EC50 = 288.7 nM T29500 CUEG14 122179430 Ki = 0.1 nM T29500 CV51WL 122179431 Ki = 29.9 nM T29500 C5PW9Y 123141715 IC50 = 835.9 nM T29500 C03AHG 123183757 IC50 = 1284 nM T29500 CK4ZO0 123183788 IC50 = 617.6 nM T29500 C17PEO 123204312 IC50 = 3266 nM T29500 C9W8OX 123311113 IC50 = 8488 nM T29500 CCK90I 123322716 IC50 = 5320 nM T29500 C8AKN7 123368349 IC50 = 866.1 nM T29500 C5I2VU 123378354 IC50 = 1361 nM T29500 C9ZCI2 123387804 IC50 = 4320 nM T29500 C6LRF9 123393714 IC50 = 4807 nM T29500 CU7CX9 123415538 IC50 = 980.5 nM T29500 C3HJV5 123437117 IC50 = 2162 nM T29500 CO3CT2 123472560 IC50 = 2197 nM T29500 C8RU2P 123475619 IC50 = 169.6 nM T29500 C8XV2H 123562321 IC50 = 70.9 nM T29500 CF2R5U 123576734 IC50 = 2248 nM T29500 C1HE3L 123644751 IC50 = 1206 nM T29500 C9IR4A 123667086 IC50 = 32.7 nM T29500 C3CK5L 123688273 IC50 = 158.5 nM T29500 CAN97K 123752717 IC50 = 3139 nM T29500 C9CO7R 123801568 IC50 = 2768 nM T29500 CI4TU7 123854385 IC50 = 287.1 nM T29500 C2T0KW 123986550 IC50 = 7583 nM T29500 C7T0GE 124018870 IC50 = 168.9 nM T29500 CM57GR 126720252 Ki = 1110 nM T29500 CTBN56 127026052 Ki < 10000 nM T29500 CU49VE 127036186 Ki = 1778.28 nM T29500 CG06BD 127036932 Ki = 794.33 nM T29500 CVW71O 127036953 Ki = 1995.26 nM T29500 CXR71M 127038002 Ki = 5.754 nM T29500 CL5N3P 127038713 Ki = 72.44 nM T29500 C89SOL 127040060 Ki = 114.82 nM T29500 CQ3L8Z 127040156 Ki = 79.43 nM T29500 CCH14Q 127041710 IC50 = 180 nM T29500 C8A1TO 127043026 IC50 > 10000 nM T29500 C3GX2A 127044893 IC50 = 5992 nM T29500 C6P4LV 127044894 IC50 = 610.2 nM T29500 C70SOF 127044906 IC50 = 2959 nM T29500 C1I6UZ 127044911 IC50 = 262.9 nM T29500 CX9PE0 127044912 IC50 = 130.6 nM T29500 CXKQ86 127044916 IC50 = 936.6 nM T29500 CL40YC 127045050 IC50 = 640.6 nM T29500 C50GOC 130442480 Ki = 8800 nM T29500 CM04RF 130442572 Ki = 7400 nM T29500 CN2KE8 131978695 IC50 = 7928 nM T29500 C7FM0U 132060763 Ki > 10000 nM T29500 CT81OY 132060776 Ki = 7330 nM T29500 CFXL21 132060812 Ki = 4890 nM T29500 C7CSU4 132075278 Ki > 10000 nM T29500 CT58QY 132578518 EC50 = 608.4 nM T29500 C8H7BY 132578519 EC50 = 42.1 nM T29500 CAVB41 132584404 Ki > 10000 nM T29500 C6D1HC 134132279 Ki > 1000 nM T29500 CQ95LB 134133571 Ki > 1995.26 nM T29500 CM4XE8 134133829 Ki = 218.78 nM T29500 CBG14F 134136412 EC50 = 104.8 nM T29500 CYXO49 134136428 EC50 = 14.15 nM T29500 CG9J7V 134136763 Ki = 50.12 nM T29500 CKH7W6 134137025 Ki = 190.55 nM T29500 C5A6XO 134138438 Ki = 407.38 nM T29500 CP67BZ 134138882 IC50 > 10000 nM T29500 CB0S8Y 134139869 Ki = 10.47 nM T29500 C3W5SM 134139893 Ki = 100 nM T29500 CHG9Z5 134140686 Ki > 1995.26 nM T29500 CFW7E3 134141385 Ki > 1995.26 nM T29500 CYW9L4 134142282 IC50 > 10000 nM T29500 C46ZTY 134143085 Ki = 549.54 nM T29500 C3NT1H 134143679 Ki > 1995.26 nM T29500 C2IM4X 134143913 Ki > 1995.26 nM T29500 C7GT5Y 134145079 IC50 > 10000 nM T29500 CXN73G 134147055 Ki = 13.8 nM T29500 C1QZ5S 134147190 IC50 = 9170 nM T29500 CS2OC5 134147929 Ki = 25.12 nM T29500 CYK0E3 134148037 EC50 = 461.1 nM T29500 C94IEA 134148920 EC50 = 12.65 nM T29500 CBU81N 134149168 Ki > 10000 nM T29500 C7HT1Z 134149596 Ki = 12.88 nM T29500 C0CEH2 134149598 IC50 > 10000 nM T29500 CEU53H 134149777 Ki = 194.98 nM T29500 C1PQ5T 134150412 Ki > 1995.26 nM T29500 C4BH9V 134150497 Ki = 77.62 nM T29500 CF46WD 134150827 IC50 > 10000 nM T29500 C3H7KF 134151231 EC50 = 598.6 nM T29500 C9IAC0 134152568 Ki = 14.79 nM T29500 CDWP64 134153527 Ki = 436.52 nM T29500 CJ45MK 134154987 EC50 = 15.5 nM T29500 CFW4O8 134156323 EC50 = 514.8 nM T29500 C6S0VM 134157330 Ki = 389.05 nM T29500 CBL29F 134157566 IC50 > 10000 nM T29500 C25RED 137631359 Ki = 251.19 nM T29500 C19JKQ 137638321 Ki = 177.83 nM T29500 CA03VC 137639125 Ki = 288.4 nM T29500 CZ4TA9 137640201 Ki = 223.87 nM T29500 CE8N4S 137641762 Ki > 10000 nM T29500 CU1O2P 137642386 Ki = 114.82 nM T29500 CKS5V0 137643541 Ki > 10000 nM T29500 CPCY48 137645406 Ki = 2173 nM T29500 C96EAP 137646245 Ki = 371.54 nM T29500 CPI68E 137646281 Ki = 94 nM T29500 CW2L7Z 137651819 Ki = 120.23 nM T29500 CR9F3Q 137653203 Ki > 10000 nM T29500 CMDV74 144096985 Ki = 44 nM T29500 CN67YQ 144096995 Ki = 30 nM T29500 C91RQY 145949210 Ki = 25.12 nM T29500 CL0XY8 145950240 Ki = 63.1 nM T29500 C45LBY 145951352 Ki = 42.66 nM T29500 CB3O4C 145951457 Ki = 177.83 nM T29500 CE3ZM8 145953314 Ki = 0.912 nM T29500 C6VO0S 145955016 Ki = 316.23 nM T29500 CT9I0G 145956955 Ki = 0.2818 nM T29500 C75KTN 145958538 Ki = 54.95 nM T29500 CX56QA 145960918 Ki = 0.7762 nM T29500 CFBX59 145962085 Ki = 46.77 nM T29500 C2FNR9 145962342 Ki = 0.1288 nM T29500 CE9I6G 145962368 Ki = 0.302 nM T29500 C0G7JA 145962478 Ki = 0.5248 nM T29500 C3DGE5 145962817 Ki = 9.12 nM T29500 C2HL4E 145962945 Ki = 1.175 nM T29500 C7BC0I 145963755 Ki = 7.413 nM T29500 C64TUP 145963761 Ki = 1100 nM T29500 CQU59F 145963832 Ki > 120 nM T29500 CZ86PI 145965488 Ki > 1200 nM T29500 C0TU9I 145965623 Ki = 880 nM T29500 CZSN84 145967270 Ki > 120 nM T29500 CBPU13 145968055 IC50 = 1124.56 nM T29500 CTJ0X5 145968736 IC50 = 583.21 nM T29500 CTP81Y 145968741 IC50 = 972.31 nM T29500 C9M7ZG 145969396 Ki > 120 nM T29500 CT9FQ7 145969986 IC50 = 672.65 nM T29500 CDLX87 145970204 IC50 = 998.17 nM T29500 C7IGH9 145970995 Ki = 430 nM T29500 CQIB05 145975238 Ki = 150 nM T29500 CF8ET9 145975365 Ki > 120 nM T29500 C0W3YR 145977627 Ki > 120 nM T29500 CC2G1V 146025727 Ki = 4800 nM T29500 C6P3SR 153287553 Ki > 10000 nM T29500 CV9G7Z 153287572 Ki > 10000 nM T29500 CO85KL 153287574 Ki > 10000 nM T29500 C7N0VH 155512508 Ki > 1000 nM T29500 C7W1OH 155513940 Ki = 91.2 nM T29500 CV8F7A 155515301 Ki = 380.19 nM T29500 CT4U8D 155517137 Ki > 1000 nM T29500 CAV5Y1 155519565 Ki > 1000 nM T29500 CUSA24 155519891 Ki > 10000 nM T29500 CL07FB 155521817 Ki > 1000 nM T29500 CXEB36 155523275 Ki > 1000 nM T29500 CYZ60F 155524736 Ki > 1000 nM T29500 CD5BI1 155525649 Ki = 102.33 nM T29500 C8GC1P 155526628 Ki = 14.79 nM T29500 CIO6V1 155528183 Ki > 1000 nM T29500 C7FR8Y 155529117 Ki = 102.33 nM T29500 CF2DM6 155529314 Ki = 25.12 nM T29500 C3ZL2V 155531279 Ki > 1000 nM T29500 C3R4YM 155532148 Ki = 22.91 nM T29500 C3MXL6 155532834 Ki = 15.85 nM T29500 CTU64O 155533099 Ki = 3019.95 nM T29500 CU3YE7 155534933 Ki > 1000 nM T29500 CB79ZW 155536080 Ki > 10000 nM T29500 CQG68A 155536202 Ki = 107.15 nM T29500 CFH7K5 155542074 Ki = 95.5 nM T29500 C91VXF 155544397 Ki > 1000 nM T29500 CR54LA 155544513 Ki = 37.15 nM T29500 CXH9A8 155549493 Ki > 1000 nM T29500 C9XQ8H 155552820 Ki = 281.84 nM T29500 C4LOH3 155555858 Ki = 30.9 nM T29500 C0CV6O 155557695 Ki = 2290.87 nM T29500 C3UCM2 155557792 Ki = 67.61 nM T29500 C20QMI 155558704 Ki > 1000 nM T29500 CE0HN5 155559841 Ki > 1000 nM T29500 C8ZKT3 155562124 Ki = 56.23 nM T29500 C71MOD 155563001 Ki = 27.54 nM T29500 C3DK0P 155565218 Ki = 165.96 nM T29500 CVU9O2 155565448 Ki = 64.57 nM T29500 C19PZX 155565707 Ki > 1000 nM T29500 CRX52O 155567200 Ki = 31.62 nM T29500 CB2VD8 44241743 Ki = 31 nM T29500 D00GEE 92766 Ki = 517 nM T29500 D01BJZ 9817640 Ki = 39.81 nM T29500 D01KAX 135453290 Ki > 30000 nM T29500 D01WWC 16573 Ki > 950 nM T29500 D02NNS 9845181 Ki = 165 nM T29500 D03DET 10287730 Ki = 1000 nM T29500 D03TPY 9885123 IC50 > 10000 nM T29500 D04BYL 10352428 Ki = 4000 nM T29500 D05EQG 5265 Ki = 7.079 nM T29500 D05GDP 599482 Ki > 10000 nM T29500 D05RWZ 6603724 Ki = 134000 nM T29500 D05XGR 6918647 Ki = 2511.89 nM T29500 D05ZUX 44207909 Ki = 910 nM T29500 D06ABL 9891980 Ki = 0.45 nM T29500 D06QKW 2765 EC50 = 63.1 nM T29500 D06UBB 123981 Ki = 485 nM T29500 D07LRJ 5312149 Ki = 1995.26 nM T29500 D07QCC 10946567 Ki = 15 nM T29500 D08CKM 9863250 Ki < 3162.28 nM T29500 D08XTL 9866614 Ki = 10000 nM T29500 D09RPR 16737207 Ki > 10000 nM T29500 D09ZUW 6603904 Ki = 2 nM T29500 D0D8GV 9830741 Ki = 119 nM T29500 D0DP8I 132266 Ki = 0.1349 nM T29500 D0EO4F 9891167 Ki = 9.09 nM T29500 D0FF6S 16038374 IC50 > 10000 nM T29500 D0H3CW 9839317 Ki = 783 nM T29500 D0H7PC 6918553 Ki > 7943.28 nM T29500 D0H9QG 5312148 Ki < 15848.93 nM T29500 D0L5MW 181743 Ki = 1191 nM T29500 D0M5ZE 5311416 Ki = 501.19 nM T29500 D0N7UE 10198248 Ki = 3235.94 nM T29500 D0O3GF 1220 Ki > 1000 nM T29500 D0O6MG 3567002 Ki = 31.62 nM T29500 D0Q4PY 9888164 Ki = 3536 nM T29500 D0Q7ZR 9890547 Ki = 4.66 nM T29500 D0T2RY 9948320 Ki = 65 nM T29500 D0V6DJ 5640 Ki = 39.81 nM T29500 D0Z7EA 643606 Ki = 0.6 nM T29500 D0Z8OD 9887378 Ki = 46120 nM T72732 C3VRO9 44557921 IC50 > 10000 nM T72732 C9WGB8 127035904 IC50 = 3300 nM T72732 D0X8BU 71718651 IC50 = 5800 nM T01269 D0MU9L 176077 IC50 = 42 nM T01269 D0S5LT 29435 Ki = 18000 nM T01269 C2P0AK 480948 IC50 = 805000 nM T01269 CX76PN 6475030 IC50 = 80000 nM T01269 C90QNU 9882222 IC50 = 9500 nM T01269 CJ6TV8 10011928 IC50 > 1000000 nM T01269 CZT1D2 10080697 Ki = 67000 nM T01269 CE9XP3 10240946 Ki > 2000000 nM T01269 CE2AF4 10352016 IC50 = 920000 nM T01269 CLKA50 11240664 IC50 = 390000 nM T01269 CJE5T9 12103482 IC50 = 14000 nM T01269 CW28RN 12103488 IC50 = 53 nM T01269 CT0JI3 13018788 IC50 = 45000 nM T01269 C40CSF 25181192 IC50 = 22100 nM T01269 CYBM80 44367875 IC50 > 1000000 nM T01269 CF7H4C 44368231 IC50 > 1000000 nM T01269 C75BDZ 44368232 IC50 > 1000000 nM T01269 CS5ZN1 44368239 IC50 = 725000 nM T01269 C1JWV2 46906966 IC50 = 224000 nM T01269 CEP1M9 90664182 Ki = 300000 nM T01269 C9SN4L 90664183 Ki = 400000 nM T01269 CVK90M 102029945 IC50 = 34200 nM T01269 C3WBY2 127025939 Ki > 2000000 nM T01269 C30RWL 127027504 Ki > 2000000 nM T01269 C9J8LD 127027505 Ki > 2000000 nM T01269 C9WSG4 137632720 IC50 = 5000 nM T01269 C2NOP7 137639289 IC50 = 7700 nM T01269 CZJT84 137641705 IC50 = 3000 nM T01269 C4EAZ0 137646452 Ki = 2000 nM T01269 CKFJ47 137656079 IC50 = 13000 nM T01269 C7YNR0 145950365 IC50 = 3500 nM T01269 CDE64Z 145951974 IC50 = 3100 nM T01269 C6M5NI 145956209 IC50 = 1200 nM T01269 C2J4TZ 145956399 Ki = 3500 nM T01269 C2M5WG 145963126 IC50 = 13000 nM T01269 CT0Q8H 145965670 IC50 = 159000 nM T01269 CXZH98 145971016 IC50 = 185000 nM T01269 CE8RL1 145972204 IC50 = 4100 nM T01269 CE40SO 145978797 IC50 = 171000 nM T01269 D07RRH 46906930 IC50 = 15000 nM T01269 D0Q1KL 44320078 IC50 = 6400 nM T01269 D0R8TR 445612 IC50 = 40000 nM T01269 D0RU5N 46906931 IC50 = 39000 nM T01269 D0SQ1T 10261406 Ki = 500 nM T67207 D0H5CD 5748217 IC50 = 40 nM T67207 D0P8YC 5362422 IC50 = 100 nM T67207 C9VJG3 9820317 EC50 = 100 nM T67207 CM97TO 9866534 IC50 = 230 nM T67207 CO8CY4 10000020 EC50 = 1400 nM T67207 CLC84V 10075168 IC50 = 16 nM T67207 CK4OG2 10321079 IC50 = 20 nM T67207 C7GK0A 10343478 IC50 = 1600 nM T67207 CS70LJ 10388253 IC50 = 600 nM T67207 CA75GC 10453674 IC50 = 20 nM T67207 CT23RH 44327170 IC50 = 200 nM T67207 C3LBS5 44327223 IC50 = 3700 nM T67207 CCY3J1 44327232 IC50 = 1900 nM T67207 C0WX4Z 44327233 IC50 > 20000 nM T67207 CP5B1W 44327235 IC50 = 5000 nM T67207 CVR1S3 44327236 IC50 = 8000 nM T67207 CP79CH 44327243 IC50 > 20000 nM T67207 CC8IX0 44327244 IC50 = 1000 nM T67207 CW14ZM 44327247 IC50 > 20000 nM T67207 CTKF67 44327298 IC50 > 20000 nM T67207 CJF81U 44327375 IC50 > 20000 nM T67207 CDL26B 44327405 IC50 = 5000 nM T67207 CRPT39 44327418 IC50 > 20000 nM T67207 C2V1BQ 44327419 IC50 > 20000 nM T67207 C94BYD 44327428 IC50 > 20000 nM T67207 C12NGR 44327430 IC50 = 5000 nM T67207 CM2E3F 44327431 IC50 > 20000 nM T67207 C4HD3I 44327475 IC50 >> 20000 nM T67207 CDGA70 44335755 EC50 = 6960 nM T67207 CY06LU 44335763 EC50 > 10000 nM T67207 CLBK94 44335776 EC50 > 10000 nM T67207 C0D1KR 44335780 EC50 = 1940 nM T67207 C51AWB 44335814 EC50 > 10000 nM T67207 C8NAL5 44335826 EC50 > 30000 nM T67207 CZ89QH 44335827 EC50 = 5600 nM T67207 CHF16Y 44335865 EC50 > 10000 nM T67207 CV3Q9W 44335875 EC50 > 10000 nM T67207 CO9K8F 44335885 EC50 = 110 nM T67207 C7Y5ZB 44335902 EC50 = 20700 nM T67207 C4WHC0 44336073 EC50 = 6300 nM T67207 CVY9W3 44336128 EC50 > 10000 nM T67207 C9A2MJ 44336147 EC50 = 3500 nM T67207 CM3F2G 44337397 IC50 = 220 nM T67207 CC2HT8 44337415 IC50 = 1000 nM T67207 CE70RM 44337427 IC50 = 100 nM T67207 CDW4I0 44337430 IC50 = 320 nM T67207 C8GR3H 44337445 IC50 = 760 nM T67207 CJ6MP1 44337450 IC50 = 100 nM T67207 C1U5YS 44337471 IC50 > 1000 nM T67207 C6VKC0 44337510 IC50 > 10000 nM T67207 C0QD2V 44337525 IC50 > 20000 nM T67207 CG63XT 44337531 IC50 > 1000 nM T67207 C9L3HU 44337570 IC50 = 20 nM T67207 CQ9PR4 44337572 IC50 > 10000 nM T67207 C5ONP9 44337593 IC50 = 80 nM T67207 CD5ZE7 44337599 IC50 = 400 nM T67207 C2TY9L 44337602 IC50 > 20000 nM T67207 CT82PD 44341747 IC50 = 20 nM T67207 C0GC5F 44341759 IC50 = 30 nM T67207 C83FUZ 44341941 IC50 = 100 nM T67207 CS69CM 44341968 IC50 = 3700 nM T67207 C5S0YH 44341969 IC50 = 100 nM T67207 CHR3Q5 44341970 IC50 = 50 nM T67207 C8LG0S 44342114 IC50 = 40 nM T67207 CD59OJ 44342127 IC50 = 30 nM T67207 C8MFA9 44342168 IC50 = 160 nM T67207 C3K2CH 44342173 IC50 = 80 nM T67207 CXWQ20 44342181 IC50 = 20000 nM T67207 CTLH31 44342210 IC50 ~ 1000 nM T67207 CP5KS3 44342211 IC50 = 130 nM T67207 CN9J4G 44342228 IC50 = 3000 nM T67207 CE1TJ7 44342237 IC50 = 1000 nM T67207 CIW84B 44342238 IC50 = 13 nM T67207 CC1JA5 44342253 IC50 ~ 100 nM T67207 C2Y3DX 44342284 IC50 = 380 nM T67207 CT3EL5 44342419 IC50 = 100 nM T67207 CG0X7W 44342441 IC50 = 210 nM T67207 C7XCR5 44342451 IC50 = 100 nM T67207 C2OL0I 71457963 IC50 = 70 nM T67207 CYB60V 71458014 IC50 = 70 nM T67207 D00EIL 6419747 EC50 = 313 nM T67207 D0R2BO 194777 IC50 = 1000 nM T02389 D00QET 5281040 IC50 = 0.43 nM T02389 D05DVP 5717 Ki = 0.3 nM T02389 D08QIP 4887 IC50 = 0.044 nM T02389 D07GTB 16760063 Ki = 0.2 nM T02389 D0B7KF 129968 Ki = 42 nM T02389 D0J4EG 122010 Ki = 6200 nM T02389 D0J7UI 115219 Ki = 0.2 nM T02389 D0O8ZE 5059 IC50 = 510 nM T02389 D0S8YL 3969 Ki = 600 nM T02389 D0ZE5V 23662025 IC50 = 100 nM T02389 CUOI21 60539 Ki = 35 nM T02389 C9T3FB 105007 IC50 = 35 nM T02389 C5SZ0H 126144 Ki = 445 nM T02389 C4W2BO 126145 Ki = 245 nM T02389 CT09PW 126778 IC50 = 10 nM T02389 CQ4XF0 128237 IC50 = 0.37 nM T02389 CK3Y9H 129044 Ki = 3 nM T02389 C5WR9V 178974 IC50 = 7.943 nM T02389 C4LNF0 178975 IC50 = 50.12 nM T02389 C0OC6D 184800 IC50 = 100 nM T02389 CZ6NE8 3082609 IC50 = 1000 nM T02389 CB0K8R 6070260 IC50 > 50000 nM T02389 CSZ5C3 6223893 IC50 = 560 nM T02389 C7K8CB 6917955 Ki = 400 nM T02389 CY9MA1 9809348 IC50 = 0.34 nM T02389 C6U9GD 9820486 IC50 = 600 nM T02389 CRH6D8 9820984 IC50 = 120 nM T02389 C53TGM 9822618 IC50 = 0.9 nM T02389 C50ESJ 9829145 IC50 = 0.19 nM T02389 C8J5BF 9829784 Ki = 0.7 nM T02389 C34ABL 9829999 IC50 = 0.54 nM T02389 CYH27W 9842487 Ki = 12 nM T02389 CJQ4C8 9868007 Ki = 60 nM T02389 CJ7QG1 9872307 IC50 = 0.9 nM T02389 C67BWX 9906952 Ki = 69 nM T02389 CUK08Y 9927762 Ki = 130 nM T02389 CH0W3D 9948371 IC50 = 200 nM T02389 C1F4WO 9948863 IC50 = 1000 nM T02389 CQ8O3D 9951001 IC50 = 2000 nM T02389 C9V1KT 9956127 Ki = 14 nM T02389 CG8J2E 10019718 IC50 = 480 nM T02389 C5Y1MZ 10074211 IC50 = 3 nM T02389 CL14HS 10381270 IC50 = 1000 nM T02389 CUI6F0 10406291 IC50 = 580 nM T02389 CLW49P 10431536 IC50 = 1500 nM T02389 CP32UQ 13019311 IC50 = 500 nM T02389 CI5K0H 13389149 IC50 = 2000 nM T02389 CU8C6Z 13389152 IC50 = 100 nM T02389 CHD50I 13389156 IC50 = 200 nM T02389 C3M9JE 13389159 IC50 = 200 nM T02389 CK56FI 13389160 IC50 = 1000 nM T02389 CYW4A3 13389161 IC50 = 100 nM T02389 CQR76T 13389163 IC50 = 200 nM T02389 C9HT2J 13389164 IC50 = 1000 nM T02389 C5N2HD 13389165 IC50 = 400 nM T02389 CZX0V2 13389166 IC50 = 500 nM T02389 CE1J7B 13505604 IC50 = 200 nM T02389 CF74OQ 13505606 IC50 = 200 nM T02389 C81XYA 13505609 IC50 = 80 nM T02389 C6XYU9 13770359 IC50 = 800 nM T02389 CVJ4Y7 13781054 IC50 = 100 nM T02389 C5IUR4 13781055 IC50 = 12.59 nM T02389 CS26UX 13781056 IC50 = 12.59 nM T02389 COX0I4 13781057 IC50 = 10 nM T02389 CM9J1B 13781058 IC50 = 12.59 nM T02389 C85DFE 13781059 IC50 = 15.85 nM T02389 C28RHG 13781060 IC50 = 39.81 nM T02389 CF9Z6Y 13781061 IC50 = 31.62 nM T02389 C7HIL1 13781062 IC50 = 19.95 nM T02389 CM2DU0 13781063 IC50 = 316.23 nM T02389 C5UOK3 13781064 IC50 = 12.59 nM T02389 CA9GB6 13781065 IC50 = 15.85 nM T02389 C9GE6S 13781066 IC50 = 19.95 nM T02389 CJ3E1M 13781067 IC50 = 50.12 nM T02389 CKJ1A7 13781068 IC50 = 100 nM T02389 CW75IO 13781069 IC50 = 630.96 nM T02389 C7IL5Q 13781070 IC50 = 10 nM T02389 CJ3DN9 13781077 IC50 = 398.11 nM T02389 C3BQ6M 13781083 IC50 = 100 nM T02389 C9TBX8 13781092 IC50 = 100 nM T02389 C68OTP 13781095 IC50 = 501.19 nM T02389 C8WJ0C 13781097 IC50 = 630.96 nM T02389 CI5AL8 13997647 IC50 = 20000 nM T02389 C0ET1F 13997651 IC50 = 9000 nM T02389 CW4XF7 13997652 IC50 = 3000 nM T02389 CG7I0Z 13997658 IC50 = 3100 nM T02389 C4F9RM 13997659 IC50 = 370 nM T02389 CJE49K 13997661 IC50 = 830 nM T02389 C5DSC4 13997662 IC50 = 30 nM T02389 C3U0QT 13997664 IC50 = 240 nM T02389 C9TK7P 13997666 IC50 = 1000 nM T02389 C4OYD7 13997667 IC50 = 300 nM T02389 C67DLF 13997668 IC50 = 32 nM T02389 C4EG9N 13997694 IC50 = 40000 nM T02389 C28PRO 13997695 IC50 = 2600 nM T02389 C6AMR9 13997696 IC50 = 1500 nM T02389 C1AB9M 13997697 IC50 = 208.93 nM T02389 CL70FW 13997698 IC50 = 70.79 nM T02389 C1IT8V 13997699 IC50 = 100 nM T02389 C9UV4I 13997700 IC50 = 158.49 nM T02389 C1KM2H 13997701 IC50 = 501.19 nM T02389 C8P1SW 13997702 IC50 = 2200 nM T02389 CPTO74 13997703 IC50 = 220 nM T02389 C76JLC 13997704 IC50 = 9400 nM T02389 CT80EG 13997705 IC50 = 5000 nM T02389 CH7J9B 13997706 IC50 = 100 nM T02389 C6S9XR 13997707 IC50 = 12.88 nM T02389 CXL7Y1 13997708 IC50 = 8.913 nM T02389 CJ84WZ 13997709 IC50 = 14.13 nM T02389 CCV98N 13997710 IC50 = 19.95 nM T02389 C9XM8Q 13997711 IC50 = 300 nM T02389 CYW6U3 13997712 IC50 = 180 nM T02389 C2GNF9 13997713 IC50 = 15.14 nM T02389 C1PQ8O 13997714 IC50 = 4.169 nM T02389 CK2P8V 13997715 IC50 = 5.495 nM T02389 C1GRH3 13997716 IC50 = 7 nM T02389 CY0DV2 13997717 IC50 = 5 nM T02389 CG51CH 13997718 IC50 = 53 nM T02389 CUDG21 13997719 IC50 = 0.8511 nM T02389 CCGL32 13997720 IC50 = 0.5 nM T02389 CJX9V1 13997721 IC50 = 5.495 nM T02389 CJ4S1A 13997722 IC50 = 7.413 nM T02389 CG36ZR 13997723 IC50 = 2150 nM T02389 CS2LD0 13997724 IC50 = 490 nM T02389 C1QV9F 13997725 IC50 = 220 nM T02389 CKYF37 13997726 IC50 = 140 nM T02389 C6BIS1 13997727 IC50 = 350 nM T02389 CQK1B4 13997728 IC50 = 580 nM T02389 CZ4N1U 13997729 IC50 = 3200 nM T02389 CZEI63 13997730 IC50 = 1100 nM T02389 CMJ43U 13997731 IC50 = 660 nM T02389 C7I8KE 13997732 IC50 = 120 nM T02389 CWY97H 13997733 IC50 = 2300 nM T02389 C1AGB3 13997734 IC50 = 150 nM T02389 C6EIW8 13997735 IC50 = 120 nM T02389 CB48TI 13997736 IC50 = 21 nM T02389 C29QKJ 13997737 IC50 = 88 nM T02389 CWJ09V 13997738 IC50 = 215 nM T02389 CCX50W 13997739 IC50 = 34 nM T02389 CV21QF 13997740 IC50 = 100 nM T02389 CLQ57T 13997741 IC50 = 18 nM T02389 CJ7FO6 13997742 IC50 = 140 nM T02389 CVN61L 13997743 IC50 = 150 nM T02389 C9RS1Y 13997744 IC50 = 4.3 nM T02389 C4ZIX8 13997745 IC50 = 0.47 nM T02389 C9HPI7 13997746 IC50 = 2 nM T02389 CN5XK6 13997748 IC50 = 5.2 nM T02389 C43QZE 13997749 IC50 = 1.3 nM T02389 CSA0R7 13997750 IC50 = 0.67 nM T02389 CL6EP2 13997752 IC50 = 1.1 nM T02389 C6BVN7 13997753 IC50 = 62 nM T02389 CW63RP 13997754 IC50 = 20 nM T02389 CGSE41 13997755 IC50 = 11 nM T02389 CJKE69 13997756 IC50 = 1.5 nM T02389 CN5OR7 13997757 IC50 = 0.031 nM T02389 CWLR63 13997758 IC50 = 0.06 nM T02389 CI05QY 13997759 IC50 = 0.11 nM T02389 C40JAW 13997760 IC50 = 0.14 nM T02389 CLT24M 13997761 IC50 = 0.16 nM T02389 CTC2O8 14097573 Ki = 1180 nM T02389 CAI73F 14097574 Ki = 5674 nM T02389 CA70PZ 14097575 Ki = 287 nM T02389 CSVN45 14097576 Ki = 4094 nM T02389 CZDO18 14097577 Ki = 1002 nM T02389 CK75WN 14097579 Ki = 78 nM T02389 C68RWY 14097580 Ki = 624 nM T02389 CBMJ32 14097581 Ki = 147 nM T02389 CU8HW9 14097582 Ki = 1958 nM T02389 C29RSB 14097583 Ki = 491 nM T02389 C7UIB3 14097584 Ki = 141 nM T02389 CM5GI1 14097585 Ki = 3149 nM T02389 CXE9A7 14097586 Ki = 579 nM T02389 CWZ5G8 14097587 Ki = 624 nM T02389 CE7A8B 14097588 Ki = 303 nM T02389 CMQ7W8 14097589 Ki = 156 nM T02389 CE56PV 14097590 Ki = 476 nM T02389 C9OW7I 14097591 Ki = 846 nM T02389 CQLT57 14329741 IC50 = 8000 nM T02389 CI5E7O 14329751 IC50 = 5000 nM T02389 CTS1K2 14329752 IC50 = 2000 nM T02389 CRNS76 14329984 IC50 = 200 nM T02389 C6M3ZP 14541262 IC50 = 7000 nM T02389 CK3Q1H 14541273 IC50 = 5000 nM T02389 C3A2PZ 14541286 IC50 = 4000 nM T02389 CE57YB 14541290 IC50 = 2000 nM T02389 CZ6WF7 14541295 IC50 = 6000 nM T02389 CH62MC 14626814 Ki = 0.8 nM T02389 C3ZHT5 14626815 Ki = 1.4 nM T02389 C2LT7Y 14626816 Ki = 0.2 nM T02389 C2VMR7 14626818 Ki = 67 nM T02389 CP76AM 14626830 Ki = 132 nM T02389 CO0U2N 14626847 Ki = 57 nM T02389 CT2WQ0 14626848 Ki = 53 nM T02389 C9A5CT 14626849 Ki = 71 nM T02389 CF54ZO 14626850 Ki = 84 nM T02389 CE8CL0 14626851 Ki = 70 nM T02389 C10LHI 14626852 Ki = 10 nM T02389 C1DN8U 14626854 Ki = 5.6 nM T02389 CI69AD 14626856 Ki = 6.8 nM T02389 C7NZ3G 14626860 Ki = 0.3 nM T02389 CG5T9C 14626862 Ki = 0.5 nM T02389 CX7G0L 14626865 Ki = 0.7 nM T02389 CS4QD5 14626867 Ki = 0.25 nM T02389 C7J2OM 14626868 Ki = 0.3 nM T02389 CD30FJ 14626869 Ki = 0.3 nM T02389 CHQZ09 14626870 Ki = 0.3 nM T02389 CCB21X 14626871 Ki = 0.3 nM T02389 COA56L 14626873 Ki = 0.3 nM T02389 CC5K3B 14626875 Ki = 0.25 nM T02389 C70VIF 14626877 Ki = 0.1 nM T02389 CCE94D 14650340 IC50 = 2000 nM T02389 CPF64H 14650341 IC50 = 800 nM T02389 CE3F4R 14650342 IC50 = 19 nM T02389 C1UD5O 14650343 IC50 = 140 nM T02389 C96MHJ 14650346 Ki = 18 nM T02389 CIDB83 14650348 IC50 = 25 nM T02389 CMN2C7 14650359 IC50 = 400 nM T02389 CSY31Z 14650381 IC50 = 250 nM T02389 CW49MO 14650383 IC50 = 275 nM T02389 CYV26P 14742699 Ki = 100 nM T02389 CDY4P3 14742700 Ki = 110 nM T02389 C49CWA 14742701 Ki = 90 nM T02389 CO3V1I 14742702 Ki = 140 nM T02389 CH02EU 14742703 Ki = 70 nM T02389 C5F8JH 14742704 Ki = 85 nM T02389 C5SNR8 14742705 Ki = 24 nM T02389 C23AWM 14742706 Ki = 43 nM T02389 C23OLK 14742707 Ki = 50 nM T02389 C4WV3R 14742708 Ki = 21 nM T02389 CTKE61 14742709 Ki = 52 nM T02389 CB8UY2 14742710 Ki = 31 nM T02389 CU6NX0 14742711 Ki = 20 nM T02389 C2O6IM 14742712 Ki = 31 nM T02389 C0UO7J 14742713 Ki = 34 nM T02389 C50ZXN 14742714 Ki = 17 nM T02389 C54KDM 14742715 Ki = 11 nM T02389 CUR9O0 14742717 Ki = 14 nM T02389 C25DOH 14742718 Ki = 8 nM T02389 CD86OB 14742719 Ki = 25 nM T02389 CMBJ07 14742720 Ki = 43 nM T02389 CLTF36 14742723 Ki = 51 nM T02389 C12LYF 14742727 Ki = 22 nM T02389 CUF6G7 14742733 Ki = 100 nM T02389 C60QFN 14742734 Ki = 15 nM T02389 CK1G9M 14742737 Ki = 25 nM T02389 CPES28 14742738 Ki = 43 nM T02389 C1W7BP 14750536 IC50 = 280 nM T02389 CZ85CW 14835274 Ki = 646 nM T02389 C6I5BR 14835275 Ki = 11526 nM T02389 CI2FK9 14835276 Ki = 4228 nM T02389 C5Y2XU 14835281 Ki = 2515 nM T02389 C85LON 14835291 Ki > 20000 nM T02389 CY2A0E 14835292 Ki = 423 nM T02389 CKML69 14884546 IC50 = 6900 nM T02389 CD15SY 15087130 IC50 = 0.96 nM T02389 C1U4XR 15290701 IC50 = 1.31 nM T02389 C1EZ6I 15290705 IC50 = 0.57 nM T02389 C31YRP 15290709 IC50 = 0.26 nM T02389 C0Z5YB 15291433 IC50 = 25 nM T02389 CSF61A 15291435 IC50 = 12.7 nM T02389 CO9HI1 15291439 IC50 = 2.7 nM T02389 CJK59F 15291441 IC50 = 2.4 nM T02389 CD1WY9 15291443 IC50 = 22.8 nM T02389 C2YWT5 15291446 IC50 = 0.5 nM T02389 CRC07E 15291450 IC50 = 194 nM T02389 CTI8N5 15291454 IC50 = 11.8 nM T02389 C0IO4H 20282989 IC50 = 300 nM T02389 CK73RD 22416853 IC50 = 2 nM T02389 C4W1ZI 22416855 IC50 = 1 nM T02389 CJ93GY 22416860 IC50 = 6 nM T02389 C4JVE7 22416873 IC50 = 2 nM T02389 CPL0I6 22416876 IC50 = 24 nM T02389 CVD18A 22416877 IC50 = 0.8 nM T02389 CO39XV 22416878 IC50 = 80 nM T02389 CT3UL6 22416879 IC50 = 4 nM T02389 CBVG49 22416883 IC50 = 6.4 nM T02389 CPT7W8 22416892 IC50 = 3 nM T02389 C37PNU 22416895 IC50 = 10 nM T02389 CQ0S1R 22416898 IC50 = 9 nM T02389 C6J7XN 22416903 IC50 = 1.4 nM T02389 CF42UC 22416910 IC50 = 4 nM T02389 CQ54DO 22416914 IC50 = 2500 nM T02389 CZ6N7H 22416923 IC50 = 0.5 nM T02389 C2GA7O 22416928 IC50 = 7.3 nM T02389 C7IK1Q 22416929 IC50 = 11 nM T02389 CDAH58 22416930 IC50 = 11 nM T02389 C9GV6E 23663990 Ki = 26 nM T02389 CQGR58 23689561 IC50 = 1430 nM T02389 CY71NK 23689562 IC50 = 270 nM T02389 CIZ9T2 23689563 IC50 = 39 nM T02389 C27DHI 23689564 IC50 = 54 nM T02389 CWZN82 23689566 IC50 = 1780 nM T02389 CYQ97A 23689567 IC50 = 495 nM T02389 CH2ES7 23689568 IC50 = 97 nM T02389 CY32BM 44281879 Ki = 17578 nM T02389 C6ROZ3 44281880 Ki = 2337 nM T02389 C3T5ZJ 44281892 Ki = 7565 nM T02389 CN1FC5 44281896 Ki = 401 nM T02389 C53CIZ 44281963 Ki = 530 nM T02389 C6HJT5 44281969 Ki = 3672 nM T02389 C0G2AE 44281989 Ki = 430 nM T02389 C7LK2U 44281998 Ki > 20000 nM T02389 CO2C5K 44282035 Ki > 20000 nM T02389 CZR7A9 44282065 Ki > 20000 nM T02389 CID72K 44282322 Ki = 934 nM T02389 CYW94C 44282323 Ki > 20000 nM T02389 C8RKT6 44282353 Ki > 20000 nM T02389 CY0DH6 44282402 Ki > 20000 nM T02389 C2C7DA 44282408 Ki = 2092 nM T02389 CD28XQ 44282414 Ki = 1009 nM T02389 C2JMO9 44282432 Ki = 187 nM T02389 C1Z3SN 44282441 Ki = 1246 nM T02389 CV62ZL 44294525 IC50 = 5000 nM T02389 CMV64J 44295696 Ki = 3 nM T02389 CZV2T7 44295931 Ki = 434 nM T02389 CPA3B9 44296051 Ki = 27 nM T02389 CP3R9O 44296079 Ki = 92 nM T02389 C4GD9Y 44296080 Ki = 19 nM T02389 CWF50E 44319586 IC50 = 10.9 nM T02389 CC5IT1 44319587 IC50 = 0.42 nM T02389 C2LRG6 44319715 IC50 = 0.48 nM T02389 CVP1U9 44319716 IC50 = 1.21 nM T02389 CC40AI 44319717 IC50 = 0.29 nM T02389 C4U6ML 44319718 IC50 = 0.44 nM T02389 CNL60U 44319774 IC50 = 1.43 nM T02389 CC49QG 44319782 IC50 > 150 nM T02389 CQ8NH0 44319783 IC50 = 3.21 nM T02389 CM0Y3J 44319827 IC50 = 0.87 nM T02389 CRQP48 44319872 IC50 = 0.65 nM T02389 CC58WV 44319977 IC50 = 1.03 nM T02389 CT3Z7O 44319978 IC50 = 1.93 nM T02389 CC5T1W 44319992 IC50 = 0.34 nM T02389 CC46HF 44320021 IC50 = 0.34 nM T02389 C81BFE 44320022 IC50 = 0.2 nM T02389 C35WBU 44349955 IC50 = 15 nM T02389 CB9SG7 44360538 IC50 = 410 nM T02389 CDCS71 44360573 IC50 = 1.2 nM T02389 CX9HR4 44360585 IC50 = 0.63 nM T02389 C1U4HZ 44360625 IC50 = 0.58 nM T02389 CDZ5V1 44360637 IC50 = 0.5 nM T02389 C0MH5O 44360640 IC50 = 0.35 nM T02389 C3F8DC 44360643 IC50 = 0.21 nM T02389 CB3PX8 44360644 IC50 = 0.74 nM T02389 C9I2GO 44360664 IC50 = 0.7 nM T02389 C49ORT 44360665 IC50 = 1.2 nM T02389 CB21JX 44360674 IC50 = 0.43 nM T02389 CRHZ26 44360675 IC50 = 0.73 nM T02389 CLY2J8 44360752 IC50 = 4.7 nM T02389 C9WI8M 44360808 IC50 = 421 nM T02389 CO6UZ0 44360844 IC50 = 2.6 nM T02389 C9W7TQ 44360858 IC50 = 0.17 nM T02389 C2KH6D 44360895 IC50 = 25.2 nM T02389 CRTI18 44360896 IC50 = 0.8 nM T02389 C27ZJP 44360897 IC50 = 2.4 nM T02389 C8TDS7 44360901 IC50 = 3.4 nM T02389 CSTM63 44360920 IC50 = 1.7 nM T02389 C6AU5H 44385730 IC50 = 200 nM T02389 CMOY36 44385933 IC50 = 0.3 nM T02389 C4JPS8 44386063 IC50 = 0.4 nM T02389 CPD01R 44386104 IC50 = 9 nM T02389 CD87RM 44386301 IC50 = 140 nM T02389 CX1ZD6 44386871 IC50 = 3900 nM T02389 C85XSL 71454546 Ki = 1380 nM T02389 CIC70Y 135408526 IC50 > 50000 nM T02389 C1X0FY 136114628 IC50 = 1584.89 nM T02389 D04CZQ 9888588 IC50 = 0.2 nM T02389 D0G7OZ 60842 Ki = 5 nM T02389 D0N7MS 5353376 IC50 = 14000 nM T02389 D0P4KL 135411330 IC50 > 50000 nM T83904 D06NVJ 936 IC50 = 1200 nM T83904 D0E3SH 6918837 Ki > 10000 nM T83904 D0MM8N 3686 IC50 = 15400 nM T83904 D0R0MW 5329102 IC50 = 122700 nM T83904 D09XIZ 11538455 Ki > 10000 nM T83904 D0E3LP 5113032 IC50 = 1000 nM T83904 D0H2UB 5361 IC50 = 1200 nM T83904 D0U3EP 445154 EC50 > 300000 nM T83904 D00PWQ 3820 IC50 > 100000 nM T83904 D00RNS 49847188 IC50 = 55000 nM T83904 D04JZE 3246390 IC50 = 13.76 ug.mL-1 T83904 D07NKC 49847118 IC50 = 21200 nM T83904 D0V2UZ 49847196 IC50 = 5710 nM T83904 CF06TE 2397 IC50 = 8300 nM T83904 CBY6Q1 2400 IC50 = 24100 nM T83904 CZ25OS 8514 IC50 = 1200 nM T83904 CJ7U9O 96455 IC50 = 74000 nM T83904 CE0AR3 189883 IC50 = 87200 nM T83904 C5B4CI 219626 IC50 = 58400 nM T83904 CAUC39 390603 IC50 = 8800 nM T83904 CLY6K3 661302 IC50 = 11500 nM T83904 CEUN62 689246 IC50 = 2187.76 nM T83904 C9J6IC 694858 IC50 = 10000 nM T83904 C0J1SW 694859 IC50 = 14700 nM T83904 CBD84H 698853 IC50 = 9800 nM T83904 C7ZNC9 703333 IC50 = 38300 nM T83904 C8MBJ9 707029 IC50 > 10000 nM T83904 CDS56V 786469 IC50 = 100000 nM T83904 C69SKR 823206 IC50 = 173000 nM T83904 CDVG93 878947 IC50 = 3467.37 nM T83904 CDR43K 883209 IC50 = 5800 nM T83904 CYTM90 883612 IC50 = 5495.41 nM T83904 C50DGO 901929 IC50 > 100000 nM T83904 CG78LK 943431 IC50 = 16800 nM T83904 CZDL61 1041898 IC50 = 1500 nM T83904 C3VBZ9 1095092 IC50 = 10400 nM T83904 CW48SO 1095867 IC50 = 3400 nM T83904 C0XD3L 1096276 IC50 = 3750 nM T83904 C4MIJ9 1096280 IC50 = 1640 nM T83904 CD7JH6 1096282 IC50 = 4720 nM T83904 CB3FJ6 1096291 IC50 = 2340 nM T83904 C1RVS5 1096292 IC50 = 140 nM T83904 C6YS9Z 1103548 IC50 = 7500 nM T83904 C2Q1DX 1104317 IC50 = 10000 nM T83904 CPI3Q1 1183101 IC50 > 50000 nM T83904 CU7ZT4 1183103 IC50 > 50000 nM T83904 CUJ7W0 1183104 IC50 = 6000 nM T83904 CLK57R 1183106 IC50 = 5500 nM T83904 CH9V7F 1183108 IC50 > 10000 nM T83904 C5DIE4 1230959 IC50 = 333000 nM T83904 CWD2T7 1258010 IC50 = 242000 nM T83904 CC8V0S 1328033 IC50 = 15500 nM T83904 CG3I2T 1336501 IC50 = 3900 nM T83904 CDZ38O 1351700 IC50 = 3800 nM T83904 C85ITY 1361238 IC50 = 5700 nM T83904 CB7I9R 1372572 IC50 > 50000 nM T83904 CB92ZQ 1372991 IC50 = 3400 nM T83904 C35ESD 1386598 IC50 = 3500 nM T83904 C4KIC0 1556677 IC50 = 3500 nM T83904 C4JD2N 2130402 IC50 > 50000 nM T83904 CX8WT2 2248572 IC50 = 2818.38 nM T83904 CBNP90 2725546 IC50 > 1000000 nM T83904 C3ZS5K 2728632 IC50 > 100000 nM T83904 C0YS5J 2743189 IC50 = 57000 nM T83904 C05STE 2796669 IC50 > 300000 nM T83904 CK8W6C 2803145 IC50 > 1000000 nM T83904 CI34AE 2803968 IC50 = 74000 nM T83904 CL59UC 2809977 IC50 > 1000000 nM T83904 C0CJS1 2812103 IC50 > 300000 nM T83904 CDUT62 2812815 IC50 > 1000000 nM T83904 C5I7WN 2817242 IC50 = 56700 nM T83904 C6KUN2 2818089 IC50 > 1000000 nM T83904 CD5WE9 2818241 IC50 > 1000000 nM T83904 CZ0S1D 2826537 IC50 > 1000000 nM T83904 CDWU19 2827646 IC50 = 38000 nM T83904 CP6M9Y 2861574 IC50 = 2630.27 nM T83904 CT1M7H 3106525 IC50 = 1744000 nM T83904 CKC72H 3154530 IC50 = 2500 nM T83904 CGB17R 3290567 IC50 > 100000 nM T83904 CFGT28 3518449 IC50 = 502800 nM T83904 C94ELI 3610426 IC50 = 8700 nM T83904 CJ0T4E 3612016 IC50 = 2770 nM T83904 CYN07M 3674592 IC50 = 200000 nM T83904 C6PA5E 3809911 IC50 = 136000 nM T83904 CL49TS 3815520 IC50 > 1000000 nM T83904 CN8F1I 3953303 IC50 = 35000 nM T83904 C8F6LZ 3994330 IC50 = 77800 nM T83904 CMJC34 4238838 IC50 > 100000 nM T83904 C1XOF7 4344009 IC50 > 1000000 nM T83904 C01KSB 5714655 IC50 > 300000 nM T83904 C35RHM 5811220 IC50 = 51000 nM T83904 CDMH70 5929343 IC50 > 1000000 nM T83904 CVC31J 6459022 IC50 > 100000 nM T83904 CC8BK0 6496838 IC50 = 482000 nM T83904 CW14PR 6496840 IC50 = 751000 nM T83904 CV7W1U 7408414 IC50 = 43000 nM T83904 C2O4YS 9324490 IC50 = 453000 nM T83904 C7L2MG 10100985 IC50 = 22000 nM T83904 CON17T 10428959 Ki = 5300 nM T83904 CY1JP2 11126879 IC50 = 16300 nM T83904 CFAC26 11345158 IC50 > 100000 nM T83904 CKM71Z 11362068 IC50 = 40000 nM T83904 C7GA9I 11639738 IC50 > 200000 nM T83904 CF7UG5 12476632 IC50 > 100000 nM T83904 C4DB8R 12761967 IC50 = 24600 nM T83904 CUS7H1 13505632 IC50 = 80000 nM T83904 CY1W2F 15701548 IC50 > 100000 nM T83904 C2NT6S 16094444 IC50 = 78300 nM T83904 CP1EX9 16094445 IC50 = 9500 nM T83904 CG1R0C 16094446 IC50 = 2800 nM T83904 CBO49G 16094447 IC50 = 2500 nM T83904 C8O2TF 16094448 IC50 > 100000 nM T83904 CU9J0V 16099336 IC50 = 195900 nM T83904 CVC9Y0 16739316 IC50 = 47000 nM T83904 CA4JG5 16805603 IC50 = 178700 nM T83904 C7KO1E 21106123 IC50 = 93000 nM T83904 CL2VP6 24180124 EC50 > 300000 nM T83904 CL4WV2 24180125 EC50 = 160 nM T83904 CQI29M 24180126 EC50 > 300000 nM T83904 CI1R0Y 24772043 IC50 = 7600 nM T83904 C4JTV2 24805828 IC50 = 20000 nM T83904 C27FPA 24805831 IC50 = 19500 nM T83904 CC9J6B 24806033 IC50 = 3400 nM T83904 C2YB1I 24806034 IC50 = 1000 nM T83904 CI9GK0 24806230 IC50 = 5200 nM T83904 CESI40 24806232 IC50 = 1500 nM T83904 CXG10R 24806233 IC50 = 5400 nM T83904 CU17BO 24806235 IC50 = 7900 nM T83904 CN02AZ 24806236 IC50 = 19700 nM T83904 C2D9IE 24806237 IC50 = 10100 nM T83904 CW8K3P 24806426 IC50 = 3200 nM T83904 CGX0M8 24806427 IC50 = 2300 nM T83904 CVHK48 24806430 IC50 = 2300 nM T83904 CI6JA8 24806431 IC50 = 2000 nM T83904 CQO10K 24806635 IC50 = 3400 nM T83904 C90FYH 24806636 IC50 = 4400 nM T83904 C9VN7K 24806638 IC50 = 9800 nM T83904 CM5G0K 24807049 IC50 = 6400 nM T83904 CCKL04 24807050 IC50 = 3100 nM T83904 CO0C2B 24807052 IC50 = 10600 nM T83904 CBD6M0 24807053 IC50 = 1500 nM T83904 CO6N3T 24822260 IC50 = 29000 nM T83904 CE73LG 24949066 IC50 = 109000 nM T83904 C9HJ0W 24949071 IC50 = 113000 nM T83904 C2DNI3 24949216 IC50 = 257000 nM T83904 CKN9H4 24949217 IC50 = 74000 nM T83904 CKRF97 24949372 IC50 = 129000 nM T83904 C78YOD 26289990 IC50 = 9600 nM T83904 CEWK45 36655700 IC50 = 109000 nM T83904 C7VNJ0 42597114 IC50 = 4300 nM T83904 CQKG76 42598460 IC50 = 6800 nM T83904 CX96NF 42617956 IC50 > 90000 nM T83904 CZ6H0F 42617970 IC50 = 20100 nM T83904 C4LDS3 42617971 IC50 = 10500 nM T83904 CTXB46 42617972 IC50 = 22200 nM T83904 C6EY0D 42617973 IC50 = 4800 nM T83904 C8XP2U 42617974 IC50 = 1000 nM T83904 CLU35R 43358881 IC50 > 100000 nM T83904 CI37UB 43358927 IC50 > 100000 nM T83904 CE42TX 43513979 IC50 = 3600 nM T83904 CCQ1R9 44138532 IC50 = 65000 nM T83904 CZ84LP 44222047 IC50 = 176 nM T83904 CVT7Q2 44418709 IC50 > 100000 nM T83904 CDRG29 44418710 IC50 = 20800 nM T83904 C2VF0Q 44418711 IC50 > 50000 nM T83904 C9C4GE 44418712 IC50 > 50000 nM T83904 C9AX2Y 44427280 IC50 = 63000 nM T83904 C3C2EX 44427282 IC50 = 99000 nM T83904 CL7VU9 44427283 IC50 = 50000 nM T83904 CA87DN 44427286 IC50 = 80000 nM T83904 C32ZEJ 44562081 IC50 = 100000 nM T83904 C7ALN6 44562084 IC50 = 105000 nM T83904 C9ESG5 44562177 IC50 = 86000 nM T83904 CYL5A7 44565975 IC50 = 9400 nM T83904 CT5CK0 44572628 IC50 = 29100 nM T83904 C7OTS3 44572662 IC50 = 44000 nM T83904 CIP65R 44572663 IC50 = 83400 nM T83904 CR9C0G 44572664 IC50 = 175000 nM T83904 C89PGZ 44572666 IC50 = 10000 nM T83904 CB9LM3 44572700 IC50 = 19900 nM T83904 C1FXJ8 44572701 IC50 = 49800 nM T83904 CV3JX8 44572702 IC50 = 151000 nM T83904 CHE05V 44572703 IC50 = 31100 nM T83904 C9QF3T 44572704 IC50 = 6900 nM T83904 C0OV2S 44572705 IC50 = 238000 nM T83904 C6NJG1 44572706 IC50 = 10600 nM T83904 C75FWN 44572767 IC50 = 7600 nM T83904 CS0GP4 44572768 IC50 = 92900 nM T83904 CST4L3 44572769 IC50 = 37400 nM T83904 C4IF8W 44572770 IC50 = 5500 nM T83904 C80SNU 44572771 IC50 = 72800 nM T83904 CC68AX 44572817 IC50 = 84600 nM T83904 C5EB9Z 44572818 IC50 = 8500 nM T83904 CCRZ09 44572819 IC50 = 16500 nM T83904 COYW18 44572820 IC50 = 3800 nM T83904 C7M1DY 44572821 IC50 = 33300 nM T83904 CM86CB 44596232 IC50 = 33000 nM T83904 CRB83V 44596233 IC50 = 25000 nM T83904 CUI98P 45029060 IC50 = 135400 nM T83904 CBZ6C3 45029061 IC50 = 33400 nM T83904 C4B1JN 45029063 IC50 = 10400 nM T83904 C6L5KB 45168044 Ki = 620 nM T83904 CB3VM2 45215438 IC50 = 21100 nM T83904 C2X7PV 45222595 IC50 = 1180 nM T83904 CD0T7F 45267626 IC50 > 100000 nM T83904 C74SOQ 45267627 IC50 > 100000 nM T83904 CU04RQ 45268494 IC50 = 72000 nM T83904 C2W8PE 45269359 IC50 > 100000 nM T83904 CL23BZ 45270178 IC50 > 100000 nM T83904 C50KMA 45270186 IC50 > 100000 nM T83904 C1FNP8 45272735 IC50 = 32000 nM T83904 C52OHP 45483031 IC50 = 15000 nM T83904 C67ICN 45486324 IC50 = 28000 nM T83904 CW67RQ 46231289 IC50 = 12300 nM T83904 CSZ4B8 46856246 IC50 = 4000 nM T83904 CMF17W 46871954 IC50 = 2400 nM T83904 C4B0WG 46871955 IC50 = 2900 nM T83904 CND7M5 46919126 IC50 = 2700 nM T83904 CK4I9Y 46919223 IC50 = 338000 nM T83904 CBG93L 46966768 IC50 = 159000 nM T83904 C3ONP1 46966788 IC50 = 114000 nM T83904 CGD5W6 46966849 IC50 = 85000 nM T83904 C08ZDE 49806788 IC50 = 4600 nM T83904 C1KG4Q 49847039 IC50 = 42500 nM T83904 CG7JA8 49847120 IC50 = 8600 nM T83904 CH3L8A 49847124 IC50 > 90000 nM T83904 CIPU14 49847186 IC50 > 90000 nM T83904 CDXA49 49847190 IC50 > 90000 nM T83904 C1W9TL 49847192 IC50 = 50600 nM T83904 C3AVR6 49847270 IC50 = 5600 nM T83904 CVN51C 49847272 IC50 > 90000 nM T83904 CDM36I 49871498 IC50 = 10400 nM T83904 CPU09F 52941276 IC50 = 7200 nM T83904 CMA1X5 52942684 IC50 = 77000 nM T83904 CKY3H8 52942750 IC50 = 129000 nM T83904 CQTG45 52943833 IC50 = 69000 nM T83904 C4GZ2T 52944947 IC50 = 223000 nM T83904 CO8TC4 52946220 IC50 = 66000 nM T83904 CDL1G9 52947355 IC50 = 9800 nM T83904 CM4SC8 52947577 IC50 = 30000 nM T83904 CWS7J9 52947608 IC50 = 3600 nM T83904 CBV42S 52947718 IC50 = 23000 nM T83904 C0UV1K 52948629 IC50 = 180000 nM T83904 C8QMO6 52949842 IC50 = 60000 nM T83904 CB43HP 53248456 IC50 = 35000 nM T83904 C5N6IW 53248458 IC50 = 43000 nM T83904 C29OGW 53248460 IC50 = 52000 nM T83904 C4JRF1 53257841 IC50 = 50800 nM T83904 CY60XC 53257842 IC50 = 10000 nM T83904 CY4RF0 53258187 IC50 = 5000 nM T83904 CU64YT 53379498 IC50 = 159100 nM T83904 CV3B4K 54669816 IC50 = 4300 nM T83904 CXOK60 54669818 IC50 = 13000 nM T83904 CLSD07 54669819 IC50 = 17000 nM T83904 CW3C4D 54757795 IC50 = 2900 nM T83904 C3Z2WI 54757796 IC50 = 13000 nM T83904 CLOI75 54757797 IC50 = 36000 nM T83904 C3TZ2B 54757798 IC50 = 2000 nM T83904 CH18SI 54757799 IC50 = 862000 nM T83904 CE1X5Z 54757800 IC50 = 31000 nM T83904 C8G7SA 54757892 IC50 = 6500 nM T83904 CG19XC 54757893 IC50 = 22400 nM T83904 C1VJ5D 54757894 IC50 = 56000 nM T83904 CQ95SY 54757895 IC50 = 27000 nM T83904 C62TLD 54757896 IC50 = 53000 nM T83904 C8SFD1 54757989 IC50 = 57200 nM T83904 CV6J3B 54757990 IC50 = 16000 nM T83904 CDI95E 54757991 IC50 = 7400 nM T83904 CE09PW 56659599 IC50 = 8900 nM T83904 C3T8YQ 56664966 IC50 = 190200 nM T83904 CKFY59 56669934 IC50 = 49900 nM T83904 CCEZ94 56673416 IC50 = 34400 nM T83904 CC7T2A 56674921 IC50 = 15600 nM T83904 C6ZD1F 56676724 IC50 = 26900 nM T83904 C2V6TE 56680039 IC50 = 12000 nM T83904 C7OBN1 56856349 IC50 = 13400 nM T83904 CH36XE 56857485 IC50 = 10420 nM T83904 CZ25SN 56935695 IC50 = 1000 nM T83904 C71BDL 57345649 IC50 = 88400 nM T83904 C32DTV 57391608 IC50 = 12800 nM T83904 C03DKB 57392691 IC50 > 90000 nM T83904 CV84RT 57395072 IC50 = 21300 nM T83904 CVDK34 57395074 IC50 > 90000 nM T83904 CCMV32 57398538 IC50 = 31900 nM T83904 C5FR8C 57398601 IC50 = 41700 nM T83904 CA9NY1 57400270 IC50 = 7850 nM T83904 CH0FE1 57403131 IC50 = 12400 nM T83904 C92ZDR 59053311 IC50 = 67 nM T83904 CE4IP3 60141294 IC50 = 4200 nM T83904 CM08ZL 60148504 IC50 = 570 nM T83904 CX57EP 60165377 IC50 > 100000 nM T83904 C02PIZ 60165378 IC50 = 74000 nM T83904 CV7JQ9 60165379 IC50 > 100000 nM T83904 C98IZK 60165380 IC50 = 24000 nM T83904 CE81YX 60165381 IC50 = 30000 nM T83904 CT1SK2 60165382 IC50 = 54000 nM T83904 C25HQM 60165383 IC50 = 4300 nM T83904 C4D6HC 60165506 IC50 = 1800 nM T83904 CA19BZ 60165642 IC50 = 1800 nM T83904 CV1YC9 60165643 IC50 = 1600 nM T83904 C9HR5A 60165644 IC50 = 3100 nM T83904 C70XDP 60165645 IC50 = 2100 nM T83904 C4AV6N 60165646 IC50 = 1400 nM T83904 CE89WD 60165647 IC50 = 2000 nM T83904 CSVW05 60165648 IC50 = 2700 nM T83904 CZ8NB6 60165794 IC50 = 1500 nM T83904 CCIV73 60165795 IC50 = 2000 nM T83904 CBY8D0 60165796 IC50 = 830 nM T83904 CTRX85 60165797 IC50 = 1100 nM T83904 C2BN5H 60165798 IC50 = 3400 nM T83904 CH10ND 60165799 IC50 = 1200 nM T83904 CBWX25 60167125 IC50 = 20000 nM T83904 C1I3MW 60167126 IC50 > 300000 nM T83904 COH2I7 60167127 IC50 = 88000 nM T83904 C6SWQ8 60167128 IC50 = 69000 nM T83904 CR3IQ7 60167129 IC50 = 23000 nM T83904 C0TO6E 60167270 IC50 > 300000 nM T83904 C43YCN 60167271 IC50 = 17000 nM T83904 C3HCS6 60167272 IC50 = 77000 nM T83904 CI9DZ5 60167273 IC50 > 100000 nM T83904 C04PIO 60167274 IC50 = 25000 nM T83904 C92UWL 60167276 IC50 = 53000 nM T83904 C5JGZ2 60167277 IC50 > 100000 nM T83904 CJ8MU4 60167418 IC50 = 38000 nM T83904 C8DA7M 60167419 IC50 > 100000 nM T83904 CCI6D7 60167420 IC50 = 83000 nM T83904 CAMB94 60167421 IC50 > 100000 nM T83904 C53FNR 60167422 IC50 = 39000 nM T83904 C4G6LE 60167423 IC50 = 40000 nM T83904 COHB83 60167424 IC50 = 57000 nM T83904 CFW8P3 66560225 IC50 = 1500 nM T83904 C5ZSJ2 66560226 IC50 = 6200 nM T83904 C6VD1X 66560309 IC50 = 10600 nM T83904 CQ6KI3 66560311 IC50 = 5500 nM T83904 CLF2W9 66560312 IC50 = 4500 nM T83904 C94IGH 66560391 IC50 = 1500 nM T83904 CWM6Z8 67523832 IC50 > 100000 nM T83904 C0LV7N 70089831 IC50 > 100000 nM T83904 C78HWC 70676483 IC50 = 11200 nM T83904 CL2J4U 70676484 IC50 = 30000 nM T83904 CDO4B9 70676622 IC50 = 12500 nM T83904 C5Y0CD 70676623 IC50 = 10800 nM T83904 C9ZA7E 70676624 IC50 = 16900 nM T83904 CSZ76Q 70676625 IC50 = 58500 nM T83904 C3DHW2 70676626 IC50 = 15900 nM T83904 CE80CA 70676627 IC50 = 22500 nM T83904 CA4PI8 70676628 IC50 = 29900 nM T83904 CJ3SZ9 70676792 IC50 = 30800 nM T83904 CNVG06 71304813 IC50 = 2.7 nM T83904 CWY4S0 71304814 IC50 = 10 nM T83904 C4BHW5 71304815 IC50 = 1.1 nM T83904 C5DPV0 71449454 IC50 = 93000 nM T83904 CB4A3W 71451254 IC50 > 100000 nM T83904 C7LB1U 71451255 IC50 > 100000 nM T83904 CG1EW3 71451256 IC50 = 60000 nM T83904 C9N8WG 71451257 IC50 = 83000 nM T83904 C8CLX3 71452171 IC50 = 10000 nM T83904 C73LSH 71453984 IC50 = 14400 nM T83904 C74QYN 71454816 IC50 > 100000 nM T83904 C8VKF9 71454817 IC50 > 100000 nM T83904 CRF65P 71458450 IC50 = 33000 nM T83904 C1O0HF 71459392 IC50 = 11700 nM T83904 CSP2D8 71461991 IC50 = 69000 nM T83904 C31MUQ 71654770 IC50 > 50000 nM T83904 CU31DP 71654771 IC50 = 1.8 nM T83904 CAM70V 71654772 IC50 = 4.4 nM T83904 CE73FM 71654773 IC50 = 6.5 nM T83904 COV26M 71654774 IC50 = 23 nM T83904 CQ1KA4 71654775 IC50 = 1400 nM T83904 CMR87Y 71654838 IC50 = 49000 nM T83904 CAD5K9 71654839 IC50 = 2800 nM T83904 CTF4Y0 71654840 IC50 = 170 nM T83904 CU46KD 71654841 IC50 = 30 nM T83904 C4RA6P 71654842 IC50 = 130 nM T83904 C3WYU5 71654843 IC50 = 740 nM T83904 C12RAH 71654909 IC50 = 16 nM T83904 COW48U 71654910 IC50 = 17 nM T83904 C4AP1G 71654911 IC50 = 53 nM T83904 C1O0ZQ 71654912 IC50 = 220 nM T83904 CC6AJ7 71654913 IC50 = 67 nM T83904 CUHV94 71654914 IC50 = 29 nM T83904 CA2EM4 71654987 IC50 = 150 nM T83904 CNU2D1 71654988 IC50 = 28 nM T83904 CU5HD4 71654989 IC50 = 300 nM T83904 CP71AF 71654990 IC50 = 130 nM T83904 CUE91W 71654991 IC50 > 50000 nM T83904 CQOW51 71654992 IC50 = 10000 nM T83904 CS0FQ4 71654993 IC50 > 50000 nM T83904 CLDB05 71655060 IC50 = 1.3 nM T83904 C6JCD7 71655061 IC50 = 10 nM T83904 CX85ID 71655062 IC50 = 4.8 nM T83904 C8TX2W 71655063 IC50 = 5.4 nM T83904 C1TC4J 71655141 IC50 = 110 nM T83904 CEIX13 71812123 IC50 = 4000 nM T83904 CB5R9X 72550523 IC50 = 11200 nM T83904 CZ57NL 72550525 IC50 = 6200 nM T83904 CQ7M9B 72550526 IC50 = 17900 nM T83904 C2MFT3 72550527 IC50 = 11800 nM T83904 CU0WX7 72550747 IC50 = 6000 nM T83904 CKMS38 72550748 Ki = 2280 nM T83904 C2R4FH 72664790 IC50 = 110200 nM T83904 CK6JB1 72664791 IC50 = 18500 nM T83904 CYZ9R7 72664892 IC50 = 99800 nM T83904 C6EFG7 73291970 IC50 = 1800 nM T83904 CMS0F6 73292335 IC50 = 2530 nM T83904 CMY90N 73292338 IC50 = 25800 nM T83904 C24SZG 73333807 IC50 = 45120 nM T83904 CD41CU 73333808 IC50 = 60340 nM T83904 CT3XY9 73333924 IC50 = 56050 nM T83904 CPLI82 73355035 IC50 = 1150 nM T83904 CRZ62F 73355036 IC50 = 14000 nM T83904 C5H9NW 75593280 IC50 = 6100 nM T83904 CCVJ76 76901487 IC50 = 7500 nM T83904 CD0LW7 76901489 IC50 = 6900 nM T83904 CY9L0J 76901682 IC50 = 6600 nM T83904 C87LDV 77461130 IC50 = 5300 nM T83904 C67MJT 77461131 IC50 = 6300 nM T83904 CR95BY 79200268 IC50 = 41200 nM T83904 C9YZ7D 84193791 IC50 = 100000 nM T83904 CF60MO 86302662 IC50 = 6100 nM T83904 CWB10X 86302663 IC50 = 11500 nM T83904 CM0UG8 86302664 IC50 = 10200 nM T83904 C6LE9I 90016528 IC50 = 10100 nM T83904 C2G9TE 90237400 IC50 = 2900 nM T83904 CRS6M4 90237652 IC50 = 2400 nM T83904 C0WS7K 90237726 IC50 = 6700 nM T83904 C30EUL 90237908 IC50 = 6300 nM T83904 C82XMB 90241301 IC50 = 3800 nM T83904 C3KM1P 90242664 IC50 = 7100 nM T83904 CUY6I1 90252695 IC50 = 4900 nM T83904 CMS75B 90342300 IC50 = 9100 nM T83904 C9BQM7 90342483 IC50 = 4700 nM T83904 CQT83E 90342533 IC50 = 9500 nM T83904 C4KS9Z 90342552 IC50 = 15900 nM T83904 COS26X 90342555 IC50 = 6800 nM T83904 C21EJX 90342675 IC50 = 13200 nM T83904 CK65LS 90342755 IC50 = 8400 nM T83904 C4ZKA9 90342767 IC50 = 19900 nM T83904 CY15NX 90342810 IC50 = 9400 nM T83904 C6I1XJ 90343001 IC50 = 15600 nM T83904 C1SWY7 90343011 IC50 = 18900 nM T83904 CL6RO5 90343086 IC50 = 9800 nM T83904 CA83DE 90343096 IC50 = 7300 nM T83904 CH0UA5 90343257 IC50 = 9500 nM T83904 C8XVT3 90645142 IC50 = 52780 nM T83904 CH1RY4 90645143 IC50 = 26850 nM T83904 CZIX41 90645144 IC50 = 60600 nM T83904 C9YIS4 90654860 IC50 = 32000 nM T83904 C76QJZ 90654861 IC50 > 200000 nM T83904 CAD9C4 90654862 IC50 > 200000 nM T83904 C9U5QY 90654863 IC50 = 68000 nM T83904 CG6Z9E 90654864 IC50 = 13000 nM T83904 C4K5NA 90655418 IC50 = 16100 nM T83904 CUX71H 90666423 IC50 = 16000 nM T83904 C3FY9T 90666424 IC50 = 11000 nM T83904 CCKT95 90666431 IC50 = 12000 nM T83904 CZ6CX5 90666432 IC50 = 6000 nM T83904 CRH54C 90666436 IC50 = 10000 nM T83904 CNO10S 90667111 IC50 = 5800 nM T83904 C37LPT 90667112 IC50 = 4900 nM T83904 CRXC93 90667113 IC50 = 1819.7 nM T83904 C7W6RL 90667114 IC50 = 2200 nM T83904 CNS07R 90668290 IC50 = 17600 nM T83904 CCR4S9 90668295 IC50 = 29800 nM T83904 C96YSH 90668297 IC50 = 100000 nM T83904 C9YB0P 90668300 IC50 = 77500 nM T83904 C5US4A 91673681 IC50 = 30500 nM T83904 CQO1F3 91673682 IC50 = 45800 nM T83904 C7D6FC 91800660 IC50 = 3600 nM T83904 C03GAW 98185391 IC50 = 21000 nM T83904 CP43XT 101884802 IC50 = 77.4 nM T83904 CSDE45 101884803 IC50 = 434 nM T83904 CW3TR5 101884804 IC50 = 436 nM T83904 C48DRM 101884805 IC50 = 489 nM T83904 CKR05E 101884807 IC50 = 811 nM T83904 CM40UV 101884808 IC50 = 48.3 nM T83904 CA15KO 101884809 IC50 = 869 nM T83904 CBJ50G 101884810 IC50 = 9800 nM T83904 CA7MT5 101884812 IC50 = 978 nM T83904 C0W1CO 101884813 IC50 = 4300 nM T83904 CH06TS 101884814 IC50 = 6290 nM T83904 C2QJB4 101884815 IC50 = 7570 nM T83904 CZ17MX 101884816 IC50 = 9700 nM T83904 C9D0ZO 101891555 IC50 = 3700 nM T83904 CZHG45 101891556 IC50 = 12200 nM T83904 C8D0QZ 102129226 IC50 = 900 nM T83904 C5BQ4L 105539861 IC50 = 210 nM T83904 C2VX8K 112499922 IC50 = 160 nM T83904 CM48HY 118283202 IC50 = 14000 nM T83904 CY2SJ0 118283203 IC50 = 8200 nM T83904 CHR58E 118283204 IC50 = 7800 nM T83904 C0Y8BI 118283209 IC50 = 20000 nM T83904 CL3X7K 118717122 IC50 = 12100 nM T83904 CY05KA 118717208 IC50 = 955 nM T83904 CZQB67 118717209 IC50 = 558 nM T83904 CZ5CB6 118718013 IC50 = 22000 nM T83904 CJ34VI 118719008 IC50 = 28000 nM T83904 CYN3C5 118719009 IC50 = 123000 nM T83904 C82BYR 118720021 IC50 = 1800 nM T83904 CHE8V0 118720022 IC50 = 9600 nM T83904 COG0Z4 118720023 IC50 = 2000 nM T83904 CV1E4C 118720036 IC50 = 28700 nM T83904 CL4X5D 118722832 IC50 = 5300 nM T83904 C1LIQ9 118722834 IC50 = 11000 nM T83904 C4QM5K 118722838 IC50 = 22000 nM T83904 C8SHR5 118722839 IC50 = 3300 nM T83904 CCF68H 118722840 IC50 = 16000 nM T83904 CU7OY4 118722841 IC50 = 6200 nM T83904 C71XIW 118722842 IC50 = 13000 nM T83904 CB7M3G 118722843 IC50 = 6300 nM T83904 C69BAG 118722844 IC50 = 42000 nM T83904 CUX3R9 118722845 IC50 = 57000 nM T83904 CP7RK4 118722846 IC50 = 12000 nM T83904 CCLI64 118722847 IC50 = 600 nM T83904 CUYG58 118731175 IC50 = 20000 nM T83904 C1GH5W 118731176 IC50 > 250000 nM T83904 C3K4BJ 118731177 IC50 = 96000 nM T83904 C3L7OM 118731178 IC50 = 83000 nM T83904 CX6UA1 118731307 IC50 > 250000 nM T83904 CNH5D3 118731308 IC50 > 100000 nM T83904 C1T6WZ 118738004 IC50 = 14800 nM T83904 CKO2H0 118738015 IC50 = 5300 nM T83904 CC3W5X 118738016 IC50 = 9000 nM T83904 CD71WH 118738018 IC50 = 7800 nM T83904 CAV76G 118738024 IC50 = 6800 nM T83904 CI2LJ9 118738026 IC50 = 1700 nM T83904 CQM08D 121231415 IC50 = 16.7 nM T83904 C1Q5HT 121304741 IC50 = 6030 nM T83904 CUL2N1 121304799 IC50 = 4070 nM T83904 CTDC10 121313542 IC50 = 9180 nM T83904 C0WR3T 121313543 IC50 = 2240 nM T83904 CBVZ57 121313551 IC50 = 9590 nM T83904 CHEX13 121313553 IC50 = 5240 nM T83904 C4LGE7 121313555 IC50 = 9570 nM T83904 CYA98N 121313557 IC50 = 2150 nM T83904 C3YC4L 121313558 IC50 = 3580 nM T83904 CZ4FA9 121313559 IC50 = 3360 nM T83904 C4X9TY 121313565 IC50 = 1650 nM T83904 C1Z3VY 121313567 IC50 = 6450 nM T83904 CPN1X5 121313571 IC50 = 10310 nM T83904 CCW46Z 121313574 IC50 = 2750 nM T83904 CCT1W9 121313577 IC50 = 1200 nM T83904 CE0MK2 121313581 IC50 = 5300 nM T83904 CO6HQ9 121313582 IC50 = 1900 nM T83904 C0D2KV 121313586 IC50 = 650 nM T83904 C49ITD 121313588 IC50 = 5790 nM T83904 C36QBA 121313590 IC50 = 5110 nM T83904 CGK35R 121313591 IC50 = 8680 nM T83904 C62BEU 121313599 IC50 = 5450 nM T83904 C64THI 121313602 IC50 = 13140 nM T83904 CD7J6S 121313603 IC50 = 4220 nM T83904 C86XNJ 121313607 IC50 = 3820 nM T83904 CU8H6S 121313616 IC50 = 12480 nM T83904 CJTF17 121313619 IC50 = 4200 nM T83904 CO08SG 121313620 IC50 = 7610 nM T83904 CHP06Q 121313623 IC50 = 9600 nM T83904 CW6KG7 121313638 IC50 = 3140 nM T83904 CCN56H 121313639 IC50 = 5530 nM T83904 CBYD01 121313641 IC50 = 7430 nM T83904 CY3KO2 121313644 IC50 = 11680 nM T83904 CG6FI5 122184875 IC50 = 5400 nM T83904 C1K9SO 122184876 IC50 = 1650 nM T83904 C0N8KM 122185658 IC50 = 5500 nM T83904 CVM95G 122186869 IC50 = 5100 nM T83904 C5ZYP0 122186870 IC50 = 1380 nM T83904 C97VZS 122186871 IC50 = 1410 nM T83904 CP5R3G 122186872 IC50 = 2380 nM T83904 CEOS03 122186873 IC50 = 650 nM T83904 C95ZQN 122186874 IC50 = 2260 nM T83904 CLO15R 122186875 IC50 = 3920 nM T83904 CML8G1 122186876 IC50 = 17800 nM T83904 C41TOB 122186877 IC50 = 11900 nM T83904 C57FWN 122186878 IC50 = 8320 nM T83904 CESR15 122186879 IC50 = 8750 nM T83904 C02XHR 122187733 IC50 = 7760 nM T83904 C5MGT9 122187734 IC50 = 810 nM T83904 C5XE4R 122187735 IC50 = 7710 nM T83904 CNIL28 122187736 IC50 = 1340 nM T83904 C9KT4V 122187737 IC50 = 14500 nM T83904 CBAG46 122187738 IC50 = 5520 nM T83904 CSU7W2 122187739 IC50 = 12000 nM T83904 C9J3MI 122187740 IC50 = 4500 nM T83904 C2NEW8 122187741 IC50 = 1510 nM T83904 CVX6G1 124155856 IC50 = 252 nM T83904 C8R1KL 124155864 IC50 = 251 nM T83904 CKU31X 124155865 IC50 = 157 nM T83904 C1VNS9 124155880 IC50 = 288 nM T83904 CI5SG4 124155887 IC50 = 13.5 nM T83904 C8D6VI 124155892 IC50 = 277 nM T83904 CE9HV7 124155894 IC50 = 133 nM T83904 CL43GB 124155906 IC50 = 28.9 nM T83904 C98FJW 124155909 IC50 = 35.4 nM T83904 CG4KQ0 124155918 IC50 = 29.7 nM T83904 C2SK7Z 124155921 IC50 = 15.7 nM T83904 CI3K8Z 124155944 IC50 = 171 nM T83904 CC6E5F 124155947 IC50 = 33.1 nM T83904 CDK5F1 124156051 IC50 = 36.8 nM T83904 C5H1WI 124156054 IC50 = 4800 nM T83904 CK10FP 124156076 IC50 = 107 nM T83904 CZ1X0F 124156082 IC50 = 102 nM T83904 CN6YV0 124156084 IC50 = 19 nM T83904 C6VX3U 124156175 IC50 = 251 nM T83904 CA47GR 124156294 IC50 = 26.7 nM T83904 C94NWB 124156297 IC50 = 111 nM T83904 CLU7F3 124156311 IC50 = 138 nM T83904 C25ACW 124156314 IC50 = 98.2 nM T83904 CC3H9B 124156319 IC50 = 104 nM T83904 C0F8RC 124156322 IC50 = 43.6 nM T83904 CH2BJ7 124156324 IC50 = 34.1 nM T83904 CC1B5Q 124156332 IC50 = 465 nM T83904 CZ43QA 124156333 IC50 = 94.7 nM T83904 CWT8L7 124156337 IC50 = 313 nM T83904 C2CIJ9 124156338 IC50 = 2050 nM T83904 CU51OV 124156339 IC50 = 15100 nM T83904 CM64KZ 124156375 IC50 = 216 nM T83904 CS8D4J 124156389 IC50 = 41.9 nM T83904 CO71HP 124156406 IC50 = 113 nM T83904 CTF86E 124156432 IC50 = 75.4 nM T83904 CH2MQ3 124156454 IC50 = 46 nM T83904 C5A1MN 124156461 IC50 = 1950 nM T83904 C4DR7M 124156464 IC50 = 28.1 nM T83904 C6Z3EX 124156466 IC50 = 580 nM T83904 CQ1D7V 124156477 IC50 = 519 nM T83904 CVG8H3 124156515 IC50 = 71.4 nM T83904 CB6WM9 124156519 IC50 = 41.8 nM T83904 C5X2EL 124156548 IC50 = 500 nM T83904 COW18T 124156563 IC50 = 23.4 nM T83904 C3R8OJ 124156568 IC50 = 46.8 nM T83904 CJ2F5B 124156573 IC50 = 151 nM T83904 CJ4C0I 124156580 IC50 = 2580 nM T83904 CF06XJ 124156582 IC50 = 235 nM T83904 CJQC71 124156591 IC50 = 572 nM T83904 C47GML 124156596 IC50 = 33.3 nM T83904 CUJ71O 124156601 IC50 = 22.9 nM T83904 CK74XR 124156666 IC50 = 29.3 nM T83904 CD83AZ 124156671 IC50 = 22.4 nM T83904 COD08A 124156677 IC50 = 437 nM T83904 C0R9GV 124156702 IC50 = 1370 nM T83904 CNT71Z 124156707 IC50 = 48.6 nM T83904 C7I1AZ 124156715 IC50 = 156 nM T83904 CZDJ49 124156728 IC50 = 193 nM T83904 CE1J6Y 124156731 IC50 = 22.7 nM T83904 COTD57 124156742 IC50 = 83.1 nM T83904 CLA01I 124156756 IC50 = 505 nM T83904 CP36XI 124156875 IC50 = 64.7 nM T83904 C9KP4E 124156885 IC50 = 4460 nM T83904 CSM9Q8 124156886 IC50 = 476 nM T83904 C2CI9E 124156887 IC50 = 450 nM T83904 CUBJ73 124156888 IC50 = 46 nM T83904 CV1R2F 124156892 IC50 = 41.5 nM T83904 CULA86 124156896 IC50 = 196 nM T83904 CFN1X9 124156913 IC50 = 47.8 nM T83904 CH9R8A 124156914 IC50 = 366 nM T83904 C4AXU0 124156920 IC50 = 546 nM T83904 C4Y8GT 124156967 IC50 = 1540 nM T83904 C2DKH0 124157048 IC50 = 4150 nM T83904 C4G2NW 124157054 IC50 = 26.3 nM T83904 CDR98I 124162056 IC50 = 44.7 nM T83904 CJ47PM 126720627 IC50 = 9000 nM T83904 CU4IC8 126843233 IC50 = 28 nM T83904 CWX3F6 127026308 IC50 = 33000 nM T83904 C3K2LH 127026309 IC50 = 164500 nM T83904 C7XP5J 127026865 IC50 = 1 nM T83904 CVDO61 127027151 IC50 = 310 nM T83904 CN7L5I 127027212 IC50 = 1330 nM T83904 C7ATZ5 127027510 IC50 = 14600 nM T83904 C8V0EX 127027798 IC50 = 19900 nM T83904 CUSA46 127027799 IC50 = 30900 nM T83904 CCE2G8 127027800 IC50 = 167700 nM T83904 C3EXR8 127027802 IC50 = 143000 nM T83904 C0KN9D 127027825 IC50 = 15000 nM T83904 CU02IS 127027826 IC50 = 400 nM T83904 C09NBE 127027828 IC50 > 100000 nM T83904 CA97HQ 127028097 IC50 = 1890 nM T83904 C76EYI 127028107 IC50 = 207000 nM T83904 CCV0J7 127028111 IC50 = 289000 nM T83904 CAV8M6 127028115 IC50 = 33000 nM T83904 C3DVH2 127028117 IC50 = 180 nM T83904 CG4JM6 127028118 IC50 = 420 nM T83904 CY2Z4B 127028119 IC50 = 260 nM T83904 COY59Q 127028120 IC50 = 9770 nM T83904 CLEG98 127028123 IC50 = 320 nM T83904 CW06FM 127028124 IC50 = 480 nM T83904 CCAD53 127028125 IC50 = 540 nM T83904 CEZ24F 127028126 IC50 = 540 nM T83904 C6KUQ9 127028440 IC50 = 45600 nM T83904 C6AZU4 127028441 IC50 = 1450 nM T83904 CN2XZ9 127028442 IC50 = 1920 nM T83904 CX9S6O 127032844 IC50 = 3.2 nM T83904 C8CV4N 127033814 IC50 = 332 nM T83904 C4J8WR 127034092 IC50 = 404.3 nM T83904 CH02OR 127034093 IC50 = 58.9 nM T83904 CJO78L 127034094 IC50 = 53.1 nM T83904 CY8TS5 127034095 IC50 = 143.6 nM T83904 C6FGW5 127034098 IC50 = 10.1 nM T83904 CCEP75 127034360 IC50 = 134 nM T83904 CZ2R6J 127035147 IC50 = 52910 nM T83904 CXR74F 127035863 IC50 = 13600 nM T83904 C3MP0W 127045459 IC50 = 22000 nM T83904 C84XPC 127048873 IC50 = 112 nM T83904 CBJD15 127049868 IC50 = 28.1 nM T83904 C7P8JZ 129883511 IC50 > 50000 nM T83904 CZ45LV 129906245 IC50 > 50000 nM T83904 CCH2T8 129906312 IC50 = 5600 nM T83904 CY8B2P 132837649 IC50 = 2920 nM T83904 CZX5Y3 132991423 IC50 = 8200 nM T83904 CA3L0T 134130520 IC50 > 200000 nM T83904 CWV34S 134130814 IC50 = 240 nM T83904 C53GIN 134131007 IC50 = 22200 nM T83904 C8WD3G 134132512 IC50 = 3900 nM T83904 C2RX4P 134132760 IC50 = 4240 nM T83904 C6C1OW 134137237 IC50 = 150000 nM T83904 CD0FX8 134139976 IC50 < 20300 nM T83904 C7P4OF 134141051 IC50 = 1500 nM T83904 CYAK84 134141382 IC50 = 890 nM T83904 C7B5KW 134142322 IC50 = 220 nM T83904 CC4Z9Q 134143263 IC50 = 2400 nM T83904 CC59HY 134144404 IC50 = 2261 nM T83904 CPKD12 134145576 IC50 = 1400 nM T83904 CN15TH 134148556 IC50 = 420 nM T83904 CDBF51 134148882 IC50 = 24300 nM T83904 C53ATF 134148970 IC50 = 1160 nM T83904 CRON29 134150759 IC50 = 480 nM T83904 C8MGQ9 134153152 IC50 = 1200 nM T83904 CZ8KH9 134155806 IC50 = 180 nM T83904 CWA81H 134433586 IC50 = 6650 nM T83904 C5I0OV 134433608 IC50 = 26302.68 nM T83904 CO2I4C 134433618 IC50 = 3388.44 nM T83904 CZA36C 134433738 IC50 = 1320 nM T83904 CHB70M 134820906 IC50 = 93325.43 nM T83904 C9YPF1 134820907 IC50 = 812.83 nM T83904 CZR65A 135397670 IC50 = 250 nM T83904 C64DLE 135397680 IC50 = 120 nM T83904 C51NFI 135420639 IC50 = 20000 nM T83904 C8F5SE 135425069 IC50 = 11000 nM T83904 CB53GJ 135443018 IC50 = 20300 nM T83904 CB5W8G 135547540 IC50 = 137400 nM T83904 CE3VW5 135659046 IC50 = 20300 nM T83904 CND1B8 135862920 IC50 = 22600 nM T83904 C98WZT 135862921 IC50 = 19200 nM T83904 C42VRW 135867743 EC50 = 16500 nM T83904 C7OP3T 135967826 IC50 = 91000 nM T83904 CO5PQ9 136236339 IC50 = 24200 nM T83904 CK5XC6 136240941 EC50 = 11600 nM T83904 CY0F6M 137226429 IC50 = 127200 nM T83904 CASC80 137632714 IC50 = 10400 nM T83904 CBN1V8 137633622 IC50 = 4250 nM T83904 CQ9W1P 137634939 IC50 = 22700 nM T83904 CBV3J5 137635796 IC50 = 970 nM T83904 C52NDJ 137636210 IC50 = 3740 nM T83904 CXL2G8 137636613 IC50 = 5610 nM T83904 CR1QZ6 137636840 IC50 = 4160 nM T83904 C1K4LG 137637623 IC50 = 2650 nM T83904 CCK4X6 137637636 IC50 = 7680 nM T83904 C2GEI3 137639254 IC50 = 1850 nM T83904 CKM4U0 137639610 IC50 = 1500 nM T83904 CAW2B6 137640314 IC50 = 16320 nM T83904 CH8TA9 137640449 IC50 = 1520 nM T83904 CKO3P5 137640529 IC50 = 2610 nM T83904 C93XOF 137641984 IC50 = 6030 nM T83904 C8YK2Z 137642096 IC50 = 580 nM T83904 CK1B0V 137643431 IC50 = 2580 nM T83904 CFG8V1 137643466 IC50 = 2430 nM T83904 CMX6G5 137643742 IC50 = 21200 nM T83904 CPK49B 137644297 IC50 = 5850 nM T83904 CI67CQ 137644426 IC50 = 3800 nM T83904 C3N7AJ 137644654 IC50 = 2500 nM T83904 C4U5WK 137644691 IC50 = 51100 nM T83904 CZMR63 137645021 IC50 = 3120 nM T83904 C5JKB3 137645160 IC50 = 3140 nM T83904 C86BKT 137646021 IC50 = 2840 nM T83904 CJY3B5 137648076 IC50 = 3090 nM T83904 C9FN7L 137649628 IC50 = 730 nM T83904 CX8VR0 137649828 IC50 = 2990 nM T83904 C3CA8J 137650068 IC50 = 6600 nM T83904 CKC1B4 137650110 IC50 = 7590 nM T83904 C8ZP3X 137650567 IC50 = 1270 nM T83904 CNMS74 137650853 IC50 = 5490 nM T83904 CSX3T7 137650908 IC50 = 19800 nM T83904 CX81MH 137653263 IC50 = 2930 nM T83904 C9YUC2 137653845 IC50 = 8150 nM T83904 CCP52Y 137654178 IC50 = 1900 nM T83904 C9Z3LK 137654291 IC50 = 1110 nM T83904 CR64PY 137654402 IC50 = 3680 nM T83904 CLBD61 137654646 IC50 = 2500 nM T83904 C9NCK7 137654659 IC50 = 4000 nM T83904 CYE1D2 137654921 IC50 = 1720 nM T83904 CL54RF 137654965 IC50 = 1830 nM T83904 CC38BQ 137654993 IC50 = 2480 nM T83904 CWZX50 137655024 IC50 = 6940 nM T83904 C9DSU1 137655468 IC50 = 2920 nM T83904 CKA2P3 137655803 IC50 = 10170 nM T83904 C7T0XQ 137655835 IC50 = 1740 nM T83904 CCYU93 137656347 IC50 = 8670 nM T83904 CJC9I8 137657467 IC50 = 2560 nM T83904 CD34PI 137657605 IC50 = 3900 nM T83904 C4FZU7 137657660 IC50 = 2600 nM T83904 C1GZ7L 137657896 IC50 = 1900 nM T83904 CIT7K5 137658301 IC50 = 49400 nM T83904 CDL6S5 137660551 IC50 = 5060 nM T83904 CLW0B7 137661474 IC50 = 390 nM T83904 C3ZY7B 137661514 IC50 = 3200 nM T83904 CU1G3C 137661872 IC50 = 3780 nM T83904 CAQ62X 137701235 Ki > 10000 nM T83904 C62HXG 138319670 IC50 = 2400 nM T83904 CN2UH1 139303146 IC50 > 20000 nM T83904 C15QPM 145949537 IC50 > 300000 nM T83904 CA3HP1 145949621 IC50 = 41300 nM T83904 CUP2O0 145950742 IC50 = 1318.26 nM T83904 C0WX7G 145950856 IC50 = 75857.76 nM T83904 CD03RC 145951020 IC50 > 300000 nM T83904 CHF0D5 145951161 IC50 = 141253.75 nM T83904 CYX85E 145951428 IC50 = 29400 nM T83904 CX4R7H 145952006 IC50 > 300000 nM T83904 CGVU43 145952074 IC50 = 173780.08 nM T83904 CJBA07 145952477 IC50 = 300000 nM T83904 C0EKS7 145952756 IC50 > 300000 nM T83904 CNL90I 145953107 IC50 > 301995.17 nM T83904 C52RBV 145953733 IC50 = 89125.09 nM T83904 CAJX35 145953758 IC50 > 300000 nM T83904 CFO9U4 145953925 IC50 = 11700 nM T83904 CN84AC 145954292 IC50 = 15135.61 nM T83904 C0DKM2 145954819 IC50 > 300000 nM T83904 C0GR1A 145956014 IC50 = 122600 nM T83904 CN6KC5 145956141 IC50 = 127700 nM T83904 C6PCI8 145956292 IC50 = 109500 nM T83904 C9PV2G 145957468 IC50 = 70794.58 nM T83904 CD0FW9 145957670 IC50 > 300000 nM T83904 CIYL61 145958186 IC50 = 168800 nM T83904 C51PDZ 145958500 IC50 > 301995.17 nM T83904 C67GPY 145958990 IC50 > 300000 nM T83904 CXM1S2 145960080 IC50 > 300000 nM T83904 CW7HG8 145960911 IC50 = 20000 nM T83904 CM76LA 145961009 IC50 > 300000 nM T83904 C53KON 145961629 IC50 = 269153.48 nM T83904 CEN5T2 145961648 IC50 > 300000 nM T83904 C5J2MW 145962276 IC50 = 141253.75 nM T83904 CC0VT3 145962411 IC50 = 35000 nM T83904 C5PT1R 145962932 IC50 = 100200 nM T83904 CCXR94 145963449 IC50 = 2300 nM T83904 CX6L7T 145963544 IC50 = 3100 nM T83904 C5QIN6 145963700 IC50 = 237000 nM T83904 CX3MQ7 145965297 IC50 = 8610 nM T83904 C9XT0U 145966202 IC50 = 46950 nM T83904 C6W3YP 145966373 IC50 = 16120 nM T83904 CHQ8Z0 145967555 IC50 = 38100 nM T83904 C7ML9P 145967841 IC50 = 310 nM T83904 CC3G2E 145970505 IC50 = 36760 nM T83904 C9CJ3Y 145971573 IC50 = 13480 nM T83904 CY12ZR 145971711 IC50 = 300000 nM T83904 CP1I5W 145972149 IC50 = 41400 nM T83904 C1QO8I 145973119 IC50 = 44450 nM T83904 C37XVC 145973165 IC50 = 9560 nM T83904 CLT69F 145975278 IC50 = 7870 nM T83904 CWD0A9 145983712 Ki > 10000 nM T83904 C56MWZ 145986208 Ki > 10000 nM T83904 C2Y1QX 153412137 IC50 = 16400 nM T83904 C8AS1P 155512143 IC50 = 1000 nM T83904 C80DBU 155512388 IC50 = 150 nM T83904 CPZ01A 155512728 IC50 = 61 nM T83904 CPQ48B 155513088 IC50 = 550 nM T83904 CM6VN5 155513154 IC50 = 44 nM T83904 C7X8HD 155514027 IC50 > 100000 nM T83904 CFD5K2 155514249 IC50 > 1000 nM T83904 CZE29G 155514745 IC50 = 10300 nM T83904 CJDA51 155516141 IC50 = 8.44 ug.mL-1 T83904 C5CXW6 155516906 IC50 = 15600 nM T83904 C7VC1F 155517856 IC50 = 580 nM T83904 CU0M1P 155518467 IC50 = 19 nM T83904 CN78HI 155519887 IC50 = 51 nM T83904 C2M5UT 155520367 IC50 = 1600 nM T83904 C09RAW 155520570 IC50 = 300 nM T83904 CR08AH 155520911 IC50 = 7500 nM T83904 CH78ST 155523405 IC50 = 1450 nM T83904 CSL6X2 155523899 IC50 = 4.05 ug.mL-1 T83904 CE2UP8 155524342 IC50 = 7.37 ug.mL-1 T83904 CX5DW8 155524630 IC50 = 5900 nM T83904 CFH1D8 155524740 IC50 = 60 nM T83904 C4HV9G 155525499 IC50 = 36 nM T83904 CY6SI4 155526052 IC50 = 190 nM T83904 CN94IG 155526713 IC50 = 36700 nM T83904 CUX8Q2 155528776 IC50 = 25100 nM T83904 C7H6XU 155528914 IC50 = 68 nM T83904 CTH59X 155529937 IC50 = 81 nM T83904 CI26ZC 155530715 IC50 = 1700 nM T83904 CX8SC4 155530876 IC50 = 400 nM T83904 C1JKR4 155531258 Ki = 68 nM T83904 C79YZH 155531505 IC50 = 11800 nM T83904 C9WNP0 155531613 IC50 = 120 nM T83904 C2TSR5 155531646 IC50 = 190 nM T83904 CI8O1S 155535583 IC50 = 370 nM T83904 C3E2LI 155536778 IC50 = 10200 nM T83904 CZ62YJ 155540163 Ki = 470 nM T83904 CPZQ17 155542821 IC50 = 2500 nM T83904 CSX51B 155544021 IC50 = 13300 nM T83904 CD5ZP1 155544168 IC50 = 6700 nM T83904 C61BTI 155545173 IC50 = 63 nM T83904 CH30TZ 155546485 IC50 > 100000 nM T83904 C3WAN0 155550829 IC50 = 2.1 ug.mL-1 T83904 C2FZ1M 155550843 IC50 > 100000 nM T83904 C0CJQ6 155552084 IC50 = 700 nM T83904 C3D7GP 155554414 IC50 = 160 nM T83904 C6FV9S 155554968 IC50 = 640 nM T83904 CUB3M2 155555283 IC50 = 1300 nM T83904 C04ZVD 155555393 IC50 = 2.55 ug.mL-1 T83904 CG7PH3 155555586 IC50 = 120 nM T83904 C1HYO4 155558607 IC50 = 13100 nM T83904 CYU68C 155558886 IC50 = 3300 nM T83904 C61LXC 155559532 IC50 = 5600 nM T83904 CLA4P7 155561544 IC50 = 20000 nM T83904 CY6G8M 155561971 IC50 = 21800 nM T83904 C7IWD4 155564228 IC50 = 36 nM T83904 C4CIL9 155564382 IC50 = 1200 nM T83904 CL4JR8 155564674 IC50 = 20400 nM T83904 C7W5BX 155568441 IC50 = 1180 nM T83904 CDB57V 155569351 IC50 = 850 nM T83904 D00LYI 135461039 IC50 = 34500 nM T83904 D02AYX 1403654 IC50 = 243600 nM T83904 D02EWM 1376646 IC50 = 49300 nM T83904 D03APP 4386 IC50 > 100000 nM T83904 D07WDQ 66541 IC50 = 14400 nM T83904 D08JPU 3501 IC50 > 100000 nM T83904 D09SUO 5269 IC50 = 112900 nM T83904 D09VTJ 441298 IC50 = 28000 nM T83904 D0D5ZL 369401 IC50 = 10000 nM T83904 D0E1QP 4262314 IC50 = 24800 nM T83904 D0E3NT 2130404 IC50 = 2800 nM T83904 D0F1KR 1376645 IC50 = 39400 nM T83904 D0F5JG 1341463 IC50 = 12500 nM T83904 D0L8HO 2399 IC50 = 4700 nM T83904 D0M5FF 5083 IC50 = 800 nM T83904 D0TO6S 2396 IC50 = 7300 nM T83904 D0UO1E 135491748 IC50 = 25900 nM T87633 D0OJ4L 3652 IC50 = 110 nM T87633 CNKJ47 11189680 IC50 = 20 nM T87633 CSZ9E8 11474810 IC50 = 2400 nM T87633 C29BUS 25105690 IC50 = 4.6 nM T87633 CRH90Q 44589003 IC50 = 5200 nM T87633 CJ53QX 44589026 IC50 = 30 nM T87633 CQAJ97 45102599 IC50 = 15 nM T87633 C9ZX1U 45137909 IC50 = 98 nM T87633 CS2C1K 54760105 IC50 = 3.9 nM T87633 CMY13U 54760109 IC50 = 8.6 nM T87633 CC20ZM 54760285 IC50 = 73 nM T87633 CC02GF 54760475 IC50 = 20 nM T87633 CRK2L3 54760476 IC50 = 3.5 nM T87633 CO3MX1 54760671 IC50 = 28 nM T87633 C9CY4L 54760856 IC50 = 13 nM T87633 CRLQ30 54761040 IC50 = 11 nM T87633 CDN2B1 54761215 IC50 = 11 nM T87633 C1C0IR 54761217 IC50 = 16 nM T87633 CQIU13 68246126 IC50 = 35 nM T87633 C1Q6EJ 68341156 IC50 = 27 nM T87633 CO7U3A 68341350 IC50 = 190 nM T87633 CH29GF 71258526 IC50 > 10000 nM T87633 CUC96E 117093964 IC50 = 120 nM T87633 C14VIC 117906466 IC50 = 120 nM T87633 CE0KL1 117906931 IC50 = 73 nM T87633 CR6UL3 117906934 IC50 = 56 nM T87633 C9VN3S 117906987 IC50 = 56 nM T87633 CGT95F 118721661 IC50 = 190 nM T87633 CLK82Y 118721662 IC50 = 84 nM T87633 C08QKE 118721945 IC50 > 1000 nM T87633 C6NTM8 130454358 IC50 = 130 nM T87633 C59JSA 130454361 IC50 = 50 nM T87633 C5DKT7 130454370 IC50 = 28000 nM T87633 C26WUT 130454401 IC50 = 500 nM T87633 C6FHY8 130454431 IC50 = 30 nM T87633 C6B9XI 130454445 IC50 = 18000 nM T87633 CIU01F 130454450 IC50 = 20 nM T87633 CHAE81 130454459 IC50 = 9400 nM T87633 CVEF58 130454467 IC50 = 10000 nM T87633 CG08CU 130454481 IC50 = 20 nM T87633 CTOG04 130454512 IC50 = 50 nM T87633 CY4JT1 130454516 IC50 = 80 nM T87633 CBE8V0 130454542 IC50 = 17000 nM T87633 C8RUV4 130454546 IC50 = 30 nM T87633 C7JNE6 130454574 IC50 = 40 nM T87633 CF06GU 130454579 IC50 = 4800 nM T87633 CBM73C 130454634 IC50 = 20 nM T87633 CXNZ71 130454680 IC50 = 240 nM T87633 CE86DQ 130454681 IC50 = 100 nM T87633 C0U4FJ 130472372 IC50 = 5500 nM T87633 CI84KG 130472422 IC50 = 40 nM T87633 C93TUC 130472439 IC50 = 20 nM T87633 C28LWH 130472440 IC50 = 30 nM T87633 C45BQH 132585194 EC50 = 5660 nM T87633 C14IYS 135545160 IC50 > 50000 nM T87633 CSJ29E 137222695 IC50 = 51000 nM T87633 C1DQ9N 137632868 IC50 = 133 nM T87633 C85BEX 137634734 IC50 = 2100 nM T87633 CD92WT 137635490 IC50 = 21000 nM T87633 C6UK4P 137640101 IC50 = 60 nM T87633 C5UP7W 137640859 IC50 = 99 nM T87633 C1UW7B 137641086 IC50 = 7000 nM T87633 C3GU9A 137642761 IC50 = 830 nM T87633 CN4T8D 137644178 IC50 = 308 nM T87633 CUIL14 137645168 IC50 = 590 nM T87633 CQ0A7B 137647183 IC50 < 50 nM T87633 C8PZN3 137647878 IC50 = 1100 nM T87633 C8LP5F 137653682 IC50 = 2560 nM T87633 C6CDH0 137659544 IC50 = 5100 nM T87633 CXZL91 137661216 IC50 < 50 nM T87633 CSUN37 137661892 IC50 = 100 nM T87633 CWZ59N 145978968 IC50 = 30 nM T87633 CJZ49S 145979394 IC50 = 10200 nM T87633 CGVS82 145986851 IC50 = 200 nM T87633 C6TV1L 145988217 IC50 = 4000 nM T87633 CZ2HG1 145989953 IC50 = 260 nM T87633 C6BMI0 145990319 IC50 = 110 nM T87633 CDQP96 145992257 IC50 = 30 nM T87633 CUG68V 145992733 IC50 = 5000 nM T38584 D07XHO 4413 Ki = 25 nM T38584 D0Y6SQ 2536 IC50 = 32000 nM T38584 C9EWY3 30744 IC50 = 820 nM T38584 CV1Y8U 33346 IC50 = 1100 nM T38584 C3O8YA 424477 IC50 = 300 nM T38584 CN2B6S 6852211 Ki = 17000 nM T38584 CRXV73 10175161 EC50 = 180 nM T38584 CUSH03 10218282 EC50 = 3100 nM T38584 CZUA50 11329402 Ki = 590 nM T38584 CB1S5N 11363919 Ki = 7100 nM T38584 CU07NO 11607091 Ki = 5500 nM T38584 COX6H8 12925732 IC50 = 6800 nM T38584 COYP35 12925854 IC50 > 50000 nM T38584 CP47XK 12925858 IC50 > 50000 nM T38584 CQF6D1 14480740 IC50 = 3000 nM T38584 CMZ05T 44324727 Ki = 54600 nM T38584 CE9I1R 44362422 Ki = 18200 nM T38584 CD2L8Z 44457054 IC50 > 50000 nM T38584 CA90QH 91827690 Ki = 480 nM T38584 C46MSP 118542774 Ki = 380 nM T38584 C20WBY 118542785 Ki = 9800 nM T38584 CI65YK 118542879 Ki = 160 nM T38584 CEH93P 118542958 Ki = 230 nM T38584 CITU59 118548755 Ki = 1100 nM T38584 CMF5R6 118548758 Ki = 880 nM T38584 C1IH2W 118548759 Ki = 2490 nM T38584 C6LZQ3 118548760 Ki = 350 nM T38584 C62ZNW 118548761 Ki = 520 nM T38584 C3WQ9D 118548776 Ki = 1080 nM T38584 CU01RP 118548813 Ki = 440 nM T38584 C7NG3I 118721642 Ki = 53 nM T38584 CTV97I 118721643 Ki = 96 nM T38584 C1NS7F 118721644 Ki = 65 nM T38584 C3OCD1 118721645 Ki = 58 nM T38584 CQK2U8 118721646 Ki = 80 nM T38584 C4HB3G 118721647 Ki = 60 nM T38584 CNP30X 118721648 Ki = 182 nM T38584 CRPV34 118721649 Ki = 12 nM T38584 CU5KB2 118721650 Ki = 21 nM T38584 CJA76N 118721651 Ki = 81 nM T38584 CS3GX9 118721652 Ki = 332 nM T38584 C0Y9EU 118721653 Ki = 56 nM T38584 CJ4FI3 118721654 Ki = 57 nM T38584 CK2QX9 118721655 Ki = 79 nM T38584 C4UYE3 118721656 Ki = 24 nM T38584 CP9L7H 118721657 Ki = 103 nM T38584 C2MI1J 118721658 Ki = 63 nM T38584 CIPY54 118721659 Ki = 17 nM T38584 CSAZ58 118728084 Ki > 50000 nM T38584 C4K6HY 118729129 Ki > 50000 nM T38584 C4MX0T 118729130 Ki > 50000 nM T38584 CUC7N1 118729131 Ki > 50000 nM T38584 C1KWF0 118729132 Ki = 22200 nM T38584 C1XVF0 118729853 IC50 = 600 nM T38584 C0S3EN 118729854 IC50 > 50000 nM T38584 CS7QD3 118729855 Ki = 10100 nM T38584 CWK9I0 118729856 Ki = 14000 nM T38584 C73DSK 118729857 Ki > 50000 nM T38584 CM2E0V 118729858 Ki = 16200 nM T38584 C63TEA 118729859 Ki = 20000 nM T38584 CPD68M 118729860 Ki > 50000 nM T38584 COY83A 122535266 Ki = 9375 nM T38584 CG5S2R 122535267 Ki = 6827 nM T38584 CAI69W 123238067 Ki = 1920 nM T38584 C76BAD 123424620 Ki = 430 nM T38584 CA30BN 127033248 Ki = 46500 nM T38584 CO7PY0 127033521 Ki > 100000 nM T38584 CE0QZ4 127033522 Ki = 39600 nM T38584 C7ZIR9 127034099 Ki = 1110 nM T38584 CD06PE 134313025 Ki = 33 nM T38584 CJP64T 155510867 IC50 = 780 nM T38584 CUP78D 155512098 IC50 > 20000 nM T38584 C1RYT8 155517297 Ki = 4303 nM T38584 CX6C5Y 155520312 IC50 = 6300 nM T38584 CE01NY 155523107 IC50 > 20000 nM T38584 CW9K3R 155523263 IC50 = 14000 nM T38584 CGMP07 155523803 Ki = 30 nM T38584 C4HN6V 155525157 Ki > 10000 nM T38584 C7SB9X 155528083 Ki = 2961 nM T38584 CG68UH 155529134 IC50 = 8600 nM T38584 CN0B2S 155529433 Ki = 4771 nM T38584 C5QT3D 155529505 Ki > 10000 nM T38584 CA82SM 155530516 Ki = 3.7 nM T38584 CER1Z8 155532768 Ki > 10000 nM T38584 C1HAW5 155533558 IC50 = 6000 nM T38584 CEFK81 155534191 Ki > 10000 nM T38584 C7M2UT 155534310 IC50 = 1200 nM T38584 C2YB0P 155535378 Ki > 10000 nM T38584 C6AE0I 155535379 Ki = 4634 nM T38584 CUV1I4 155535874 IC50 > 20000 nM T38584 CT4S3M 155544624 IC50 > 20000 nM T38584 C5FZ3I 155545003 Ki = 3197 nM T38584 CA08GE 155545013 Ki = 963 nM T38584 CQ51DI 155546002 IC50 > 20000 nM T38584 CK0E7M 155548720 IC50 = 18000 nM T38584 C3R9TO 155551160 IC50 = 9000 nM T38584 CM3X6Y 155555703 Ki = 6122 nM T38584 CXYR84 155556203 Ki = 1208 nM T38584 CM63SG 155557605 IC50 > 20000 nM T38584 C0IW5Z 155557962 IC50 = 8800 nM T38584 C3VJ5W 155559076 Ki = 7984 nM T38584 CY60RV 155559158 Ki = 468 nM T38584 CQ3MJ4 155559840 Ki = 8634 nM T38584 C0B3ID 155562970 Ki > 10000 nM T38584 CTF0S7 155566456 Ki = 7.2 nM T38584 D08KCA 72429 Ki = 188 nM T08722 D00NAX 4926 EC50 = 5000 nM T08722 D01ZII 2726 EC50 = 2000 nM T08722 D04MSM 2554 EC50 > 10000 nM T08722 D06ZUK 3696 EC50 = 10000 nM T08722 D09EGZ 2719 EC50 = 4000 nM T08722 D0D1AL 3559 EC50 > 10000 nM T08722 D0T2XU 4927 EC50 = 8000 nM T08722 C71OQJ 4757 EC50 > 10000 nM T08722 C78ENM 6077 EC50 = 5000 nM T08722 D0O2DQ 237 EC50 = 300 nM T53612 C03HVZ 7665603 IC50 = 15000 nM T53612 CNZA87 9112697 IC50 = 43000 nM T53612 CSP20T 10623756 IC50 > 30000 nM T53612 C35WAX 10624280 IC50 = 8200 nM T53612 C2W4YZ 10695208 IC50 = 7750 nM T53612 CZ7FS4 16284785 IC50 = 9000 nM T53612 C56TPZ 16285203 IC50 = 10000 nM T53612 C1KZB9 16289649 IC50 = 170000 nM T53612 C0YLF9 18392346 IC50 = 2900 nM T53612 C5N8IA 35192951 IC50 > 200000 nM T53612 CX05JF 38330775 IC50 = 4400 nM T53612 CS9TK6 38335241 IC50 = 130 nM T53612 CU5YR1 41583852 IC50 = 640 nM T53612 CW5V7Y 44559839 IC50 = 13500 nM T53612 C5MX2D 57404340 IC50 = 890 nM T53612 CT97OB 134405495 IC50 = 6200 nM T53612 CMNH75 134405503 IC50 = 28000 nM T53612 C2IV8D 134405509 IC50 = 23000 nM T53612 CI5Z8V 134405578 IC50 = 17000 nM T53612 CIT83E 134405671 IC50 = 58000 nM T53612 CW9NJ0 134415778 IC50 <= 2.5 nM T53612 CST8A1 134415837 IC50 = 18 nM T53612 CDQ62V 137637214 Ki > 50000 nM T53612 C2K8JV 137639385 Ki > 50000 nM T53612 CNX46H 137654508 Ki > 50000 nM T53612 CN8Q9C 137701230 IC50 = 250 nM T53612 C4JOB0 145964839 IC50 = 100 nM T53612 C5UEF9 145964989 IC50 = 130 nM T53612 CZ4UG0 145965461 IC50 = 13000 nM T53612 CPX49F 145965710 IC50 = 6990 nM T53612 C5OW8S 145965790 IC50 = 7600 nM T53612 C6FVD9 145965959 Ki = 1500 nM T53612 C7FBM1 145966386 IC50 > 200000 nM T53612 C9GFI6 145966669 IC50 = 190 nM T53612 CZ0T4L 145966695 IC50 = 490 nM T53612 CJBG50 145967253 IC50 > 50000 nM T53612 C68DYZ 145967534 IC50 = 290 nM T53612 CG6JM2 145969172 IC50 = 1200 nM T53612 C8WC0H 145971850 IC50 = 1400 nM T53612 C0IYB7 145972755 IC50 > 200000 nM T53612 CEW8K6 145974663 IC50 = 100 nM T53612 C6EOB1 145974963 IC50 = 8900 nM T53612 C5IKH6 145975051 IC50 = 2310 nM T53612 C8RY7N 145975239 IC50 = 250 nM T53612 C1RHV5 145976020 IC50 = 2800 nM T53612 C3BY5K 145976653 IC50 = 7500 nM T53612 C5P1GV 145977162 IC50 = 6000 nM T53612 CXC5Q4 145977795 IC50 = 150 nM T53612 CZ2YC3 145977988 IC50 = 110000 nM T53612 C5L2MD 145978027 IC50 = 1200 nM T53612 D00HWJ 18392356 IC50 = 1500 nM T53612 D00KJP 10322586 IC50 > 30000 nM T88452 D00YWP 9904 Ki = 724.44 nM T88452 D00ZFP 5870 Ki = 10000 nM T88452 D04DJN 10635 Ki = 1202.26 nM T88452 D06XMU 6013 Ki = 190.55 nM T88452 D07BSQ 5994 Ki = 41.69 nM T88452 D08QMX 5757 Ki = 10000 nM T88452 D0B4RU 8955 Ki = 5888.44 nM T88452 D0D1SG 5755 Ki = 30.9 nM T88452 D0I1LH 5839 Ki = 524.81 nM T88452 D0K0EK 5881 Ki = 10000 nM T88452 D0KR5B 5754 Ki = 13.18 nM T88452 D0Z1FX 5756 Ki = 10000 nM T88452 D0H5HO 5879 Ki = 2454.71 nM T88452 D08DZZ 10634 Ki = 10000 nM T88452 C2Y8WA 5744 Ki = 28.18 nM T88452 C29SPL 5867 Ki = 128.82 nM T88452 CV1Z6A 11687 Ki = 562.34 nM T88452 CMFE70 94166 Ki = 165.96 nM T88452 C3CW4N 101674 Ki = 1584.89 nM T88452 CLUP61 101773 Ki = 10000 nM T88452 CD1PN3 151150 Ki = 20.42 nM T88452 C1GY4B 228864 Ki = 151.36 nM T88452 C4RG3T 242332 Ki = 10000 nM T88452 C0C7IY 44325375 Ki = 75.86 nM T88452 D03TNT 5753 Ki = 13.18 nM T88452 D04SQY 6166 Ki = 22.39 nM T88452 D06WBH 6238 Ki = 18.2 nM T88452 D09MWG 5880 Ki = 5888.44 nM T88452 D0GW2Y 440707 Ki = 13.18 nM T88452 D0M8RO 6128 Ki = 1737.8 nM T59577 CG2PZ0 1072066 IC50 = 330 nM T59577 CX85QO 1072081 IC50 = 74.13 nM T59577 C4D2QB 36294314 IC50 = 32 nM T59577 CD1O3L 36295259 IC50 = 7 nM T59577 CKQ26F 39572558 IC50 = 39.81 nM T59577 CEFG97 86579897 IC50 = 2934 nM T59577 CRG9V0 86579900 IC50 = 21 nM T59577 C7I8VA 86579902 IC50 = 19.05 nM T59577 CCF2W7 86579937 IC50 = 28.84 nM T59577 CF1AZ9 86579938 IC50 = 23.99 nM T59577 CUJ41Q 86579939 IC50 = 17 nM T59577 CIT1M4 86579940 IC50 = 31 nM T59577 CJAT04 86579941 IC50 = 97.72 nM T59577 C82JOV 86579942 IC50 = 67.61 nM T59577 CAR82N 86579981 IC50 = 19 nM T59577 CSM2L4 86579982 IC50 = 16.98 nM T59577 CA39NC 86579984 IC50 = 12.88 nM T59577 CQ4WP2 86579985 IC50 = 43.65 nM T59577 CZT25M 86580332 IC50 = 28 nM T59577 CO29AN 90655990 IC50 = 18.2 nM T59577 C9JSK7 90655991 IC50 = 15.85 nM T59577 CQD4Y2 90655992 IC50 = 5 nM T35824 D05VZE 119031 IC50 = 10000 nM T35824 D0T9HG 132519 IC50 = 8 nM T35824 CJS23I 9868333 Ki > 5554 nM T35824 CG38KL 9936728 Ki = 107 nM T35824 CR7T3J 10009978 Ki > 2000 nM T35824 CR5H6E 10163627 Ki > 5554 nM T35824 CK0P3F 10186536 Ki > 5454 nM T35824 C4K1MJ 10208262 Ki > 5554 nM T35824 C6WZ4F 10367355 IC50 = 22 nM T35824 CFKA79 10395015 Ki = 2000 nM T35824 C5WV1N 10439082 Ki > 2000 nM T35824 C1IW7N 11292680 IC50 = 51 nM T35824 C8C5AV 11294179 Ki > 10000 nM T35824 C02BWA 11967143 Ki > 2000 nM T35824 CS46XU 16126723 IC50 = 11.4 nM T35824 CB7V8Y 25147773 IC50 = 0.31 nM T35824 C3KF1V 25178145 IC50 = 1 nM T35824 CEP9Q2 25180867 IC50 = 1.56 nM T35824 C7U1YC 25181080 IC50 = 44 nM T35824 C85HLG 25181081 IC50 = 186 nM T35824 CHR2P1 25183768 Ki > 25000 nM T35824 CT80ED 44219901 IC50 = 15000 nM T35824 C9T5ZF 44220093 IC50 = 5000 nM T35824 CLRT69 44247751 IC50 = 32 nM T35824 CGQ92A 44364037 IC50 = 56 nM T35824 C36YLM 44364111 IC50 = 202 nM T35824 CN4T7Q 44364119 IC50 = 177 nM T35824 CH4TE7 44364121 IC50 = 35 nM T35824 CPE91Y 44364122 IC50 = 21 nM T35824 CG2X0C 44364224 IC50 = 184 nM T35824 C1F8XN 44364249 IC50 = 16 nM T35824 CWM47H 44364250 IC50 = 40 nM T35824 C0W5TL 44364251 IC50 = 4633 nM T35824 C3TPO7 44364266 IC50 = 1839 nM T35824 CJ2B8F 44364280 IC50 = 1677 nM T35824 CG0Z7I 44478924 IC50 = 6000 nM T35824 CFO27Y 44478926 IC50 = 130 nM T35824 CBZJ29 44478927 IC50 = 130 nM T35824 CRJ24K 44479197 IC50 = 150 nM T35824 CGOH82 44479198 IC50 = 6500 nM T35824 CLV56M 44479199 IC50 = 730 nM T35824 CY92OQ 44479458 IC50 = 110000 nM T35824 CH1QG9 44479459 IC50 = 1200 nM T35824 CB1NT7 44479460 IC50 = 220 nM T35824 C0JQ9L 44479699 IC50 = 470 nM T35824 C0DN1Q 44479700 IC50 = 93000 nM T35824 CTG24W 44479702 IC50 = 6300 nM T35824 CGZ49M 44479703 IC50 = 1100 nM T35824 CAK94X 44563337 IC50 = 996 nM T35824 C2B0GI 45268787 IC50 = 51 nM T35824 CMPE63 45482676 IC50 = 18000 nM T35824 CU2SX3 51355576 Ki > 10000 nM T35824 CKJ9S1 56835167 IC50 = 39 nM T35824 C21CLZ 56835168 IC50 = 2200 nM T35824 C0L2TS 56835169 IC50 = 1100 nM T35824 D05THD 44478925 IC50 = 5100 nM T35824 D07GEL 10344307 Ki = 35 nM T35824 D07MJD 44479701 IC50 = 4300 nM T35824 D0A0FY 44479457 IC50 = 31000 nM T35824 D0A4TC 446504 IC50 = 6.8 nM T35824 D0H6CK 10160968 Ki > 5554 nM T35824 D0L4EO 11609208 IC50 = 32040 nM T35824 D0Q4TA 10044321 IC50 = 900 nM T35824 D0S9OL 10155934 IC50 = 1300 nM T35824 D0W2UK 6914621 Ki = 1599 nM T71949 D00SUC 74766595 IC50 = 820 nM T71949 CWJ0U1 5312 IC50 = 570 nM T71949 C06WZQ 222878 IC50 = 250 nM T71949 COS62U 245007 IC50 > 100000 nM T71949 C0MHV8 252439 IC50 = 430 nM T71949 C76AMR 439391 IC50 = 106000 nM T71949 CT0H6S 439939 IC50 = 48000 nM T71949 C2OS3W 2238068 IC50 > 100000 nM T71949 CEQ4V8 2723716 IC50 > 100000 nM T71949 C4C0EB 2816189 EC50 = 900 nM T71949 CW2JY7 5715254 Ki = 420 nM T71949 CCYF63 9942424 IC50 = 3981.07 nM T71949 CF47JU 25138011 IC50 = 4800 nM T71949 C2DBN5 46899607 IC50 = 200 nM T71949 CL3HT1 71449736 IC50 = 9100 nM T71949 CJH86V 71451542 IC50 = 3700 nM T71949 CH38AO 71453382 IC50 = 63000 nM T71949 C2U4AQ 71458738 IC50 = 370 nM T71949 C5XA3R 71733941 Ki = 11.3 nM T71949 C4PW1L 71734037 IC50 = 420 nM T71949 C14GIV 71735687 IC50 = 8000 nM T71949 CM02VN 71735839 IC50 = 9600 nM T71949 C4WS1H 71735840 IC50 = 2900 nM T71949 CT4YO5 71735841 IC50 = 16000 nM T71949 C2ZFM8 71735842 IC50 = 15000 nM T71949 CI5W0K 71735843 IC50 = 6800 nM T71949 CN5B4O 73352277 IC50 = 8100 nM T71949 C68RKH 76310231 IC50 = 7800 nM T71949 CO1EN3 76317452 IC50 = 220 nM T71949 CT5FZ8 76321184 IC50 = 12000 nM T71949 C6XRT0 76321186 IC50 = 12200 nM T71949 CKB5O9 76328366 IC50 = 12000 nM T71949 CUNK03 76335652 IC50 = 8200 nM T71949 C2NA5I 91801131 IC50 = 5011.87 nM T71949 CP3DK0 96607511 IC50 = 1200 nM T71949 C10RDJ 101882871 IC50 = 63.1 nM T71949 C86LNW 101882872 IC50 = 3162.28 nM T71949 C6NUD0 118718072 IC50 = 9100 nM T71949 C75JVN 122191451 IC50 = 12589.25 nM T71949 C3YX7W 122191453 IC50 = 31622.78 nM T71949 C3IBR8 122191455 IC50 = 6309.57 nM T71949 C59KNQ 122191457 IC50 = 10000 nM T71949 CM5X8J 122191459 IC50 = 7943.28 nM T71949 C7ASR0 122191460 IC50 = 6309.57 nM T71949 CRI6J4 122191461 IC50 = 7943.28 nM T71949 CAS4H6 122191462 IC50 = 6309.57 nM T71949 C9J6LX 122191463 IC50 = 7943.28 nM T71949 C75NJO 122191464 IC50 = 7943.28 nM T71949 C50VYK 122191465 IC50 = 3981.07 nM T71949 CSKY20 122191466 IC50 = 2511.89 nM T71949 CS3L8H 122191467 IC50 > 100000 nM T71949 CZ2NV1 122191468 IC50 = 79432.82 nM T71949 CYTW93 122191469 IC50 = 50118.72 nM T71949 CZV45H 122191470 IC50 = 5011.87 nM T71949 CF6I2N 122191471 IC50 = 6309.57 nM T71949 CZU02B 122191472 IC50 = 10000 nM T71949 CE27AS 122191473 IC50 = 12589.25 nM T71949 C87YEC 122191474 IC50 = 398.11 nM T71949 CAJ28B 122191475 IC50 = 1000 nM T71949 CQ04FW 122191477 IC50 = 12589.25 nM T71949 C12OHA 122191478 IC50 = 7943.28 nM T71949 CL2K0J 122191479 IC50 = 5011.87 nM T71949 CT6HG3 122191480 IC50 = 125.89 nM T71949 CK7LD6 122191481 IC50 = 1995.26 nM T71949 CMJ72N 122191482 IC50 = 630.96 nM T71949 C6H2YQ 122383780 IC50 = 34000 nM T71949 CT2UZ4 125377518 IC50 > 100000 nM T71949 CF7KD3 127030402 Ki = 280 nM T71949 CT4O5U 135567037 IC50 = 91000 nM T71949 CC4H1N 135567038 IC50 = 76000 nM T71949 CQBH95 135567040 IC50 > 100000 nM T71949 CP6IH9 135567041 IC50 = 89000 nM T71949 C8HMG2 135567042 IC50 = 89000 nM T71949 CL9ZD4 135567108 IC50 = 13400 nM T71949 CDY98J 135567110 IC50 = 6740 nM T71949 C1VAI3 135567112 IC50 = 8600 nM T71949 C8LFY7 135567115 IC50 = 2400 nM T71949 C34LUV 137175094 IC50 = 12900 nM T71949 C93YUK 137175210 IC50 = 2400 nM T71949 CYG29R 138393334 IC50 = 1420 nM T71949 CNG82D 138393336 IC50 = 4500 nM T71949 CARJ34 138753212 IC50 = 12540 nM T71949 C4M1EO 155519111 IC50 = 4680 nM T71949 CP8K5E 155540290 IC50 = 3770 nM T71949 CIM7D4 155548682 IC50 > 50000 nM T71949 CFR06L 155551969 IC50 > 50000 nM T71949 C3SQ4A 155569285 IC50 = 1970 nM T71949 D07IOY 10365 IC50 = 4100 nM T71949 D08IZY 3080614 IC50 = 45000 nM T71949 D0B2WZ 15331 IC50 = 1500 nM T71949 D0X5US 459617 IC50 = 15000 nM T19011 D03GET 4055 IC50 = 19000 nM T19011 C8JV3A 24465 IC50 = 30000 nM T19011 C2B6EK 752982 IC50 = 40000 nM T19011 C5MQP8 852158 IC50 > 100000 nM T19011 CI87JW 1001784 IC50 = 11000 nM T19011 CFR61E 1307198 IC50 = 9400 nM T19011 CQW6F7 1308005 IC50 = 8200 nM T19011 C7M4ID 1895639 IC50 = 5000 nM T19011 CO9ST2 2446135 IC50 = 31500 nM T19011 COE91V 2742421 IC50 = 8800 nM T19011 C7JO4Q 2820003 IC50 = 9700 nM T19011 C12CHL 4470793 Ki > 300000 nM T19011 C4VM8J 9173830 IC50 = 16800 nM T19011 CP3AO9 9356353 IC50 = 18000 nM T19011 CZ93IR 9356454 IC50 = 14200 nM T19011 CF79QB 9421427 IC50 = 47600 nM T19011 CY15NS 9880546 IC50 = 5600 nM T19011 C6YF5L 9918081 Ki > 3000 nM T19011 C6C9DL 10055263 Ki > 300000 nM T19011 CC30ZA 10305301 Ki = 178000 nM T19011 C0D9QX 10372989 Ki > 30000 nM T19011 CQO97K 10621802 IC50 = 6500 nM T19011 CRX3C7 10801994 IC50 > 80000 nM T19011 C5A3WY 11200445 IC50 = 40000 nM T19011 CQJ07W 11299775 IC50 > 100000 nM T19011 CU4E2B 11391905 IC50 > 100000 nM T19011 C3LF8B 11483880 IC50 = 3900 nM T19011 CP04UL 11484750 IC50 = 4000 nM T19011 CRPL64 11516963 IC50 = 61700 nM T19011 CSC25V 14149682 IC50 = 53900 nM T19011 CY3JU7 14646108 IC50 > 100000 nM T19011 CU8J6A 16126459 IC50 = 8600 nM T19011 C8CSM3 16126550 IC50 = 5700 nM T19011 C29ZMK 16126551 IC50 = 12600 nM T19011 C3TPL7 16126552 IC50 = 4300 nM T19011 C4Z6BF 17483715 IC50 = 10200 nM T19011 C04GYC 17531735 IC50 = 24300 nM T19011 CX42CP 17554676 IC50 = 24700 nM T19011 C12GAZ 21145366 Ki > 30000 nM T19011 CTXH84 23104907 IC50 = 20700 nM T19011 C5O0SV 24204784 IC50 > 100000 nM T19011 C7YN6L 44318744 IC50 > 2000000 nM T19011 CF3R6Y 44336593 Ki > 30000 nM T19011 CO3Z4G 44396132 IC50 > 80000 nM T19011 C0IKG2 44396147 IC50 > 80000 nM T19011 CTJZ35 44396156 IC50 > 80000 nM T19011 CBJU37 44396161 IC50 > 80000 nM T19011 CFL13J 44396193 IC50 > 80000 nM T19011 CE2A5V 44396205 IC50 > 80000 nM T19011 CU1AY3 44396206 IC50 > 80000 nM T19011 CKUR40 44396211 IC50 > 80000 nM T19011 C7RX2C 44396219 IC50 > 80000 nM T19011 CX28MD 44406938 IC50 = 2270 nM T19011 C4VO7S 44407055 IC50 > 10000 nM T19011 C0S8RA 44424744 IC50 > 100000 nM T19011 C9SJ3O 44424745 IC50 = 8800 nM T19011 CE4PU6 46873799 IC50 = 49000 nM T19011 C9FW7G 46946067 IC50 = 26000 nM T19011 C79JDN 52941554 IC50 = 5400 nM T19011 C6QCU0 52942665 IC50 = 67000 nM T19011 C73QHN 52943900 IC50 = 72000 nM T19011 CB4U2R 52945119 IC50 > 150000 nM T19011 CG3TM0 52948739 IC50 = 47000 nM T19011 CE94WN 54587113 IC50 = 50000 nM T19011 CJ2ZQ7 71697056 IC50 = 2300 nM T19011 CS76KU 90666197 IC50 = 44400 nM T19011 C96RMI 90666198 IC50 = 8600 nM T19011 CZ50TY 90666200 IC50 > 100000 nM T19011 CM92PW 121344571 IC50 <= 9000 nM T19011 CRFQ07 124165614 Ki = 400 nM T19011 C2V7NL 135797380 IC50 > 100000 nM T19011 C27EYJ 135797381 IC50 > 100000 nM T19011 CZOL36 135797386 IC50 > 100000 nM T19011 CBX75S 135797387 IC50 > 100000 nM T19011 C2L6UZ 135797388 IC50 = 56700 nM T19011 C0S1VO 135797389 IC50 > 100000 nM T19011 CS40TI 135797392 IC50 > 100000 nM T19011 C0RJW6 135797397 IC50 = 44100 nM T19011 C5UL0V 135955126 IC50 > 100000 nM T19011 C85VGD 136069445 IC50 > 100000 nM T19011 CQ7L2H 136254273 IC50 > 100000 nM T19011 C5C1XF 136254274 IC50 > 100000 nM T19011 CL4A5E 136254275 IC50 > 100000 nM T19011 CH7N3Z 136254276 IC50 > 100000 nM T19011 CL4ZM7 136254277 IC50 > 100000 nM T19011 CAHC90 136254278 IC50 = 47100 nM T19011 CQ84LN 136254279 IC50 > 100000 nM T19011 CBEU97 136254280 IC50 > 100000 nM T19011 C3LK1C 136254281 IC50 = 78200 nM T19011 C3AY7U 137631699 IC50 = 300 nM T19011 COA4K6 137632835 IC50 = 980 nM T19011 C9A6MY 137632994 IC50 = 4460 nM T19011 C2MTQ4 137633618 IC50 = 5720 nM T19011 C2K0GE 137636105 IC50 = 690 nM T19011 CL1HE3 137641758 IC50 = 800 nM T19011 CO71IL 137643613 IC50 = 14900 nM T19011 C30XET 137646265 IC50 = 5500 nM T19011 CKU6O7 137648500 IC50 = 400 nM T19011 C5DKW8 137650422 IC50 = 1440 nM T19011 C15EWQ 137653741 IC50 = 100 nM T19011 C4E9QK 137654526 IC50 = 4670 nM T19011 CQW02T 137656106 IC50 = 1000 nM T19011 CU9E1R 137656483 IC50 = 7120 nM T19011 CD2JY1 137658569 IC50 = 3640 nM T19011 CWE7I3 137659432 IC50 = 4370 nM T19011 CVO34Q 137659449 IC50 = 770 nM T19011 CNMJ89 138911333 Ki = 1900 nM T19011 CB2D3K 139600304 IC50 = 90 nM T19011 C8V0XS 155512987 Ki = 4000 nM T19011 CCQ48F 155531806 IC50 = 420 nM T19011 C4D5MV 155543902 IC50 = 210 nM T19011 D0J1KH 262093 IC50 = 78 nM T80276 D09XZB 123631 IC50 > 50000 nM T80276 D0B3HD 2519 IC50 = 400000 nM T80276 D0E6XR 3062316 IC50 = 38000 nM T80276 D0EG1I 9926791 IC50 > 10000 nM T80276 D0F8RA 2153 IC50 = 300000 nM T80276 D0J5VR 11625818 IC50 = 306.4 nM T80276 D0R0MW 5329102 IC50 = 11000 nM T80276 D0RU0O 50905713 IC50 = 1602 nM T80276 D0S5LD 135565596 IC50 = 0.5 nM T80276 D0W5HK 216239 IC50 > 50000 nM T80276 D01PGR 16123056 IC50 = 39 nM T80276 D01QSO 16654980 Ki = 20 nM T80276 D03BHZ 52913813 IC50 = 35 nM T80276 D03DPZ 45375953 Ki = 28 nM T80276 D03EZE 25167777 IC50 = 0.04 nM T80276 D03FOP 68947304 IC50 = 33000 nM T80276 D03KAC 1893730 IC50 = 39 nM T80276 D03LWG 53235510 IC50 > 9000 nM T80276 D03XAQ 49784945 IC50 = 14 nM T80276 D05EXN 58298316 IC50 = 4000 nM T80276 D06GUA 49784002 IC50 = 5011.87 nM T80276 D07BGC 57384863 Ki = 2 nM T80276 D07EHV 44814409 IC50 > 9100 nM T80276 D07HPJ 11476171 IC50 > 9100 nM T80276 D08QGT 17755052 Ki = 2.6 nM T80276 D0AW5T 9849735 IC50 = 88 nM T80276 D0C3ZR 10427712 IC50 = 1300 nM T80276 D0D8JB 44516953 IC50 = 0.4 nM T80276 D0E6UZ 54575456 IC50 = 69 nM T80276 D0H9DA 54761306 IC50 > 30000 nM T80276 D0I3LO 91933883 IC50 = 17 nM T80276 D0N5JZ 25033539 Ki = 0.57 nM T80276 D0O1IM 58298318 IC50 = 850 nM T80276 D0O1LD 11647372 IC50 = 12 nM T80276 D0O6VZ 25254071 IC50 = 4.8 nM T80276 D0TU7B 58507717 Ki = 17 nM T80276 D0U3DP 46912230 IC50 = 16 nM T80276 D0U3EP 445154 IC50 = 250 nM T80276 D0U8QH 59239165 IC50 = 4200 nM T80276 D0UP1Z 51001932 Ki = 0.29 nM T80276 D0VG0D 11977753 IC50 = 4 nM T80276 D0W7HE 56649450 IC50 = 5 nM T80276 D0X7IN 11978790 IC50 = 4 nM T80276 D0XD4I 118502708 IC50 = 320 nM T80276 D0Y2NS 70798655 IC50 = 15 nM T80276 D03BNU 59604787 IC50 > 3000 nM T80276 D05HIJ 135565159 IC50 = 1539 nM T80276 D09SFV 3973 IC50 = 300 nM T80276 D0D0QA 44137675 IC50 = 870 nM T80276 D0K1VK 25262965 IC50 = 3600 nM T80276 D0P1JI 312145 IC50 = 1 nM T80276 C3Q8HY 13205 IC50 = 20000 nM T80276 C8YU9Z 95415 IC50 = 1170000 nM T80276 CQ3LV1 124337 IC50 = 1 nM T80276 C3FRX9 131989 IC50 = 25000 nM T80276 CD7F9H 246708 IC50 = 2660000 nM T80276 CVG7P8 586366 EC50 = 196000 nM T80276 CR16JO 592738 EC50 = 79300 nM T80276 CY3D4G 617191 IC50 = 8063 nM T80276 CS5O7B 622000 IC50 > 40000 nM T80276 CXC3V1 622262 IC50 = 1333 nM T80276 CC58WG 659595 IC50 = 40000 nM T80276 CU73NO 736009 IC50 > 83300 nM T80276 CRU9G4 796828 EC50 = 170400 nM T80276 CH5QF8 1018277 IC50 = 2800 nM T80276 C3KPX5 1270546 IC50 > 20000 nM T80276 CT2VP9 1471775 IC50 = 17378.01 nM T80276 C9LG0N 1476679 IC50 > 1000000 nM T80276 C4WFP1 1587957 IC50 > 30000 nM T80276 CWOQ49 1627922 IC50 = 400 nM T80276 C9EUD2 1839691 IC50 = 10200 nM T80276 CAN89K 2762479 IC50 = 36000 nM T80276 C56YDF 2762944 IC50 = 51000 nM T80276 C09VKD 2816900 IC50 = 43200 nM T80276 C4DK0F 2819874 Ki = 230 nM T80276 C79PDA 2823822 IC50 = 1400 nM T80276 CX5E3I 2898075 IC50 = 1290000 nM T80276 CO03RG 2906609 EC50 > 500000 nM T80276 C61MCV 3100191 IC50 = 1300 nM T80276 CGHV04 3602063 IC50 = 730000 nM T80276 CBA6W9 3840028 IC50 = 40000 nM T80276 C7VW2O 4160026 IC50 = 910000 nM T80276 C1O4KS 4416330 IC50 = 2200 nM T80276 CX3IY7 4583262 EC50 = 35200 nM T80276 CIN5F7 4904109 IC50 <= 10000 nM T80276 C1YJM9 4912089 IC50 = 83000 nM T80276 CE74CV 5059890 IC50 = 100000 nM T80276 C9U2YK 5109813 IC50 = 12589.25 nM T80276 CSKN96 5350938 EC50 > 500000 nM T80276 CYQ0A1 5407855 EC50 = 139600 nM T80276 C2OZ0W 6484194 IC50 = 27600 nM T80276 CK2IR4 6852165 IC50 = 200000 nM T80276 CY01OB 9209612 IC50 = 64000 nM T80276 CE1Y8A 9815659 IC50 = 10000 nM T80276 CNQJ46 9867340 IC50 = 2.7 nM T80276 CJ79RC 9879653 IC50 = 19 nM T80276 CC4F8I 10021687 IC50 = 2700 nM T80276 CZM84H 10066542 IC50 = 2000 nM T80276 CZ15SC 10125446 IC50 = 3600 nM T80276 C2W9ED 10269329 IC50 = 500 nM T80276 C7SFI1 10296883 IC50 > 10000 nM T80276 C32NQS 10357196 IC50 = 529 nM T80276 CYRV48 10405525 IC50 = 56 nM T80276 C72LGO 10432948 IC50 = 1410 nM T80276 CAZT53 10475366 IC50 = 31 nM T80276 CL8YE3 11230964 IC50 = 3800 nM T80276 C8Y6IM 11234514 IC50 = 64 nM T80276 CT3VP7 11398307 IC50 = 3250 nM T80276 CK65NF 11418892 Ki = 50 nM T80276 CL3Z4O 11419728 Ki = 2130 nM T80276 CYBD21 11428504 IC50 = 640 nM T80276 CHJ30L 11492951 IC50 = 4500 nM T80276 CV8J3I 11514586 IC50 = 630 nM T80276 CTXF73 11515474 IC50 = 1250 nM T80276 C0O4SQ 11522078 IC50 = 330 nM T80276 C7HMO6 11526786 IC50 = 64 nM T80276 C15XPT 11529859 IC50 = 545 nM T80276 C5KV8L 11530037 IC50 = 1350 nM T80276 C1YZM3 11532472 IC50 = 44 nM T80276 CGK17J 11536358 IC50 = 185 nM T80276 C0CIM7 11539769 IC50 = 7 nM T80276 C38YWS 11541283 IC50 = 2.1 nM T80276 C1VA4C 11543481 IC50 = 3000 nM T80276 C4T8IQ 11550986 IC50 = 1800 nM T80276 C63TOQ 11551198 IC50 = 500 nM T80276 CN2MS6 11562853 IC50 = 501.19 nM T80276 CPXS32 11566902 IC50 = 600 nM T80276 CMVQ43 11576772 IC50 = 1.6 nM T80276 CX92QM 11581007 IC50 = 210 nM T80276 CEHZ82 11599141 IC50 = 316.23 nM T80276 CL5F3Z 11601890 IC50 = 190 nM T80276 C58QVA 11601930 IC50 = 455 nM T80276 C1ZPM5 11630874 IC50 = 940 nM T80276 CLK3Y4 11638999 IC50 = 100 nM T80276 CQIX52 11645168 IC50 = 1000 nM T80276 C08DUS 11645350 IC50 = 20000 nM T80276 CC64OJ 11652531 IC50 = 220 nM T80276 CP04JC 11666231 IC50 = 2.6 nM T80276 C89VFO 11669062 IC50 = 10 nM T80276 C3BT1M 11702204 IC50 = 100 nM T80276 CY8C9P 11751126 IC50 = 72 nM T80276 CBR6D5 11955693 IC50 = 290 nM T80276 CFZO21 11979157 IC50 = 7 nM T80276 C60DBM 11998444 IC50 = 23800 nM T80276 C5FTB0 11998445 IC50 = 1900 nM T80276 C68WMR 11998447 IC50 = 8393 nM T80276 CYL24B 11998448 IC50 = 2494 nM T80276 CNPI54 11998563 IC50 = 2555 nM T80276 C6AK0Y 11998564 IC50 = 3492 nM T80276 CMVA72 11998565 IC50 = 229 nM T80276 CJ3YP8 11998685 IC50 = 833 nM T80276 CV8PB5 11998690 IC50 = 676 nM T80276 CB9T1H 11998803 IC50 = 1555 nM T80276 C59SKD 11999032 IC50 = 199 nM T80276 CT58GS 12171624 IC50 = 880 nM T80276 CH52FJ 13939416 EC50 = 242000 nM T80276 CX81RT 13939417 EC50 = 335500 nM T80276 CZU1L3 14320027 IC50 = 880000 nM T80276 CY7A0T 14638904 IC50 = 8600 nM T80276 CVN8B2 16049456 IC50 = 501.19 nM T80276 C41OGY 16049526 IC50 = 260 nM T80276 CW5FD8 16081736 IC50 = 2429 nM T80276 C0I8DK 16222214 IC50 = 7200 nM T80276 CKJV37 16222216 IC50 > 10000 nM T80276 C2XW1C 16222322 IC50 = 5200 nM T80276 CP5G6J 16456450 IC50 = 162 nM T80276 CP45ET 16645457 IC50 = 970000 nM T80276 CV9US5 16736978 IC50 = 8900 nM T80276 C72THB 16739368 IC50 = 3.6 nM T80276 CF6JS9 16757570 IC50 = 23 nM T80276 CB19TH 16757576 IC50 = 4500 nM T80276 C9BJ7Q 16757577 IC50 = 2 nM T80276 C1NZC7 16757579 IC50 > 10000 nM T80276 C7TDC6 16801460 IC50 = 359 nM T80276 CEF64U 17599247 IC50 > 30000 nM T80276 CY0S6G 17751063 IC50 = 165 nM T80276 C1SN9M 17756679 IC50 >= 100000 nM T80276 CTF23G 20644743 IC50 > 100000 nM T80276 CZT32J 20877898 IC50 = 699 nM T80276 CZ0IM9 20877907 IC50 = 108 nM T80276 C0MAL8 20877967 IC50 = 1000 nM T80276 CZ7V8L 21048651 IC50 > 100000 nM T80276 C9WDR1 21270142 EC50 = 36800 nM T80276 C5UND9 21270203 EC50 = 98200 nM T80276 CVDL81 22036885 IC50 = 0.12 nM T80276 C61ZGT 22135435 IC50 > 50118.72 nM T80276 CP05ZB 22346757 IC50 = 12000 nM T80276 C1F2TM 23582995 IC50 = 4070 nM T80276 C0EJK3 23585071 IC50 = 26300 nM T80276 CEYL29 23585510 Ki = 1890 nM T80276 COW91A 23586721 IC50 = 4900 nM T80276 CVIJ28 23630332 IC50 < 2 nM T80276 CBL37C 23642173 Ki = 150 nM T80276 C8J1SI 23642272 IC50 = 2372 nM T80276 CNU8G0 23797298 EC50 > 500000 nM T80276 C29SFI 24768579 IC50 = 1972 nM T80276 CJUK39 24770517 IC50 > 10000 nM T80276 C72BSE 24804168 IC50 = 15848.93 nM T80276 CBS5J4 24804985 IC50 = 562.34 nM T80276 C6Y5GV 24805152 IC50 = 562.34 nM T80276 C9PA0M 24807809 IC50 = 1110 nM T80276 C5E4QN 24807810 IC50 > 10000 nM T80276 C3QKS1 24807976 IC50 = 66 nM T80276 CGJ60P 24807978 IC50 = 382 nM T80276 CIPF03 24808145 IC50 = 7850 nM T80276 C2XLC5 24808146 IC50 > 10000 nM T80276 C7DX6N 24808147 IC50 = 440 nM T80276 CY61FQ 24808148 IC50 = 635 nM T80276 C72QHP 24808149 IC50 = 496 nM T80276 CBMA95 24808336 IC50 > 10000 nM T80276 C7FD1B 24808337 IC50 = 638 nM T80276 CL4C8H 24809743 IC50 = 800 nM T80276 CCP2M3 24822704 IC50 > 50000 nM T80276 CP4G9Z 24855584 Ki = 110 nM T80276 CM9C0R 24866805 IC50 = 12000 nM T80276 C8E9DQ 24880629 IC50 > 83300 nM T80276 C13QYB 24884503 IC50 > 2000 nM T80276 CLX07H 24888752 IC50 = 8.6 nM T80276 CFYJ16 24888918 IC50 = 41 nM T80276 C9TO8N 24888922 IC50 = 77 nM T80276 CL78TE 24889090 IC50 = 170 nM T80276 CTS46Z 24889091 IC50 = 230 nM T80276 C57INS 24889437 IC50 > 50000 nM T80276 CFNC21 24889602 IC50 > 50000 nM T80276 COYK94 24889603 IC50 > 50000 nM T80276 C17SXC 24889765 IC50 = 49 nM T80276 CY36AQ 24889936 IC50 = 33 nM T80276 CF23RG 24889937 IC50 = 240 nM T80276 CY2W9P 24890272 IC50 = 300 nM T80276 CC01XM 24890625 IC50 = 1220 nM T80276 CPQ4Z9 24890804 IC50 = 340 nM T80276 CB79YC 24905143 IC50 = 480 nM T80276 C2DC9J 24905144 IC50 = 1100 nM T80276 CN6V8Z 24905145 IC50 = 46 nM T80276 CSB7P5 24905148 IC50 = 6300 nM T80276 CGSF21 24905149 IC50 = 9600 nM T80276 CVDG02 24905150 IC50 = 10400 nM T80276 CWH6C5 24905152 IC50 = 17 nM T80276 C0HE2Q 24905153 IC50 = 17 nM T80276 C7QSC9 24905154 IC50 = 3000 nM T80276 CO9D0K 24905155 IC50 = 1400 nM T80276 C5W9UR 24905157 IC50 = 1100 nM T80276 CC1DA3 24905158 IC50 = 1600 nM T80276 COW79F 24905159 IC50 = 1600 nM T80276 CFPA53 24905160 IC50 = 4600 nM T80276 C2O0JX 24905161 IC50 = 13700 nM T80276 CA72BE 24905162 IC50 = 1000 nM T80276 CQN6X9 24905163 IC50 = 3400 nM T80276 CD4O1F 24905165 IC50 = 3400 nM T80276 CKL48T 24905166 IC50 = 10000 nM T80276 C76VYL 24905167 IC50 = 2900 nM T80276 C7K5PU 24905168 IC50 = 1250 nM T80276 CZ57ID 24905169 IC50 = 3200 nM T80276 C2DHX9 24905170 IC50 = 7600 nM T80276 CSB96E 24905171 IC50 = 50000 nM T80276 CWZ0R2 24905172 IC50 = 2200 nM T80276 CY3B6M 24905175 IC50 = 543 nM T80276 CW1V0H 24905177 IC50 = 100000 nM T80276 CO6Y0L 24905178 IC50 = 100000 nM T80276 C60NQW 24905179 IC50 = 1910 nM T80276 C4MO8B 24905180 IC50 = 2010 nM T80276 COJI47 24905181 IC50 = 1270 nM T80276 CS0B2C 24905182 IC50 = 266 nM T80276 C1H4BT 24905183 IC50 = 520 nM T80276 C4WHK9 24905184 IC50 = 6310 nM T80276 C7Q4MZ 24905185 IC50 = 2560 nM T80276 CS4IP1 24905186 IC50 = 802 nM T80276 C69QWO 24905187 IC50 = 100000 nM T80276 C85ANB 24905188 IC50 = 652 nM T80276 CNHD75 24905189 IC50 = 289 nM T80276 C9JUO2 24905190 IC50 = 9850 nM T80276 CPR03K 24905191 IC50 = 3040 nM T80276 CTAG19 24905193 IC50 = 531 nM T80276 C7VJM5 24905194 IC50 = 1950 nM T80276 CEP1L3 24905195 IC50 = 1060 nM T80276 CP68ZD 24905196 IC50 = 2690 nM T80276 C8Z0RJ 24905197 IC50 = 813 nM T80276 CN9RT0 24905198 IC50 = 3400 nM T80276 CHI78P 24905200 IC50 = 2800 nM T80276 CO6PE8 24905201 IC50 = 2600 nM T80276 CZ63HS 24905202 IC50 = 120 nM T80276 C2X0FC 24905203 IC50 = 69 nM T80276 C0WCE3 24905204 IC50 = 35 nM T80276 CNK50B 24905205 IC50 = 70 nM T80276 C12DPB 24905206 IC50 = 82 nM T80276 C8N0RH 24905207 IC50 = 100000 nM T80276 CYA5G2 24905208 IC50 = 462 nM T80276 CDV2B4 24905209 IC50 = 1800 nM T80276 CEFK68 24905210 IC50 = 91 nM T80276 CUFP12 24905211 IC50 = 1800 nM T80276 C0JG8L 24905212 IC50 = 4000 nM T80276 CP47MK 24905213 IC50 = 19000 nM T80276 CB61QC 24905214 IC50 = 12000 nM T80276 CQ13ZI 24905215 IC50 = 32000 nM T80276 C6VI8F 24905216 IC50 = 800 nM T80276 CXNH25 24905217 IC50 = 443 nM T80276 C2PN9S 24905218 IC50 = 206 nM T80276 C9O2AL 24905219 IC50 = 752 nM T80276 CIT7U8 24905220 IC50 = 15000 nM T80276 CMD26S 24905221 IC50 = 642 nM T80276 C4R8WC 24905222 IC50 = 831 nM T80276 C47SHA 24905223 IC50 = 145 nM T80276 C1DY2R 24905224 IC50 = 209 nM T80276 CS0XF9 24905225 IC50 = 1700 nM T80276 CG5VX2 24905226 IC50 = 100000 nM T80276 C57QEO 24905227 IC50 = 100000 nM T80276 C7CG5E 24905228 IC50 = 467 nM T80276 CHP5D1 24905229 IC50 = 2400 nM T80276 CXP09S 24905230 IC50 = 344 nM T80276 CY7XG1 24905231 IC50 = 2800 nM T80276 C7JFQ2 24905232 IC50 = 245 nM T80276 C2JM1P 24905233 IC50 = 5100 nM T80276 CC3BF0 24905234 IC50 = 6800 nM T80276 CE57FI 24905235 IC50 = 2700 nM T80276 CUP20O 24905236 IC50 = 47000 nM T80276 CLC6Q2 24905237 IC50 = 3000 nM T80276 C9M1GI 24905238 IC50 = 1400 nM T80276 CVD72F 24905239 IC50 = 193 nM T80276 CK38IZ 24905240 IC50 = 86 nM T80276 CO2V5E 24905241 IC50 = 2200 nM T80276 CZBA19 24905244 IC50 = 144 nM T80276 CQ8OI1 24905246 IC50 = 100000 nM T80276 C5URC6 24905247 IC50 = 5000 nM T80276 C03SVO 24905250 IC50 = 8500 nM T80276 CIF2J5 24905251 IC50 = 1500 nM T80276 CPTE58 24905252 IC50 = 3740 nM T80276 CX1JB8 24905253 IC50 = 4200 nM T80276 COZ3H7 24905254 IC50 = 15000 nM T80276 CDT1H9 24905255 IC50 = 9000 nM T80276 C54QKA 24905256 IC50 = 4100 nM T80276 C9U0JA 24905259 IC50 = 14000 nM T80276 CO4YS7 24905260 IC50 = 17000 nM T80276 CEG0B5 24905261 IC50 = 100000 nM T80276 C9VE5F 24905262 IC50 = 100000 nM T80276 C3I4HK 24905264 IC50 = 17000 nM T80276 C0VMI6 24905265 IC50 = 100000 nM T80276 CWE3V0 24905267 IC50 = 100000 nM T80276 CH4T3A 24905268 IC50 = 100000 nM T80276 C6QDN7 24905271 IC50 = 5600 nM T80276 C6XHJ7 24905272 IC50 = 4800 nM T80276 CTB9A3 24905273 IC50 = 100000 nM T80276 C0NB1Q 24905274 IC50 = 33000 nM T80276 C9KQ0L 24905275 IC50 = 9300 nM T80276 C9O8QZ 24905277 IC50 = 4900 nM T80276 CP50RD 24905280 IC50 = 187 nM T80276 CG13ZM 24905281 IC50 = 650 nM T80276 CF0S6X 24905282 IC50 = 620 nM T80276 C5HBL0 24905284 IC50 = 14700 nM T80276 C2Z5DN 24905285 IC50 = 1500 nM T80276 CL6GH8 24905286 IC50 = 705 nM T80276 CKYO98 24905287 IC50 = 280 nM T80276 CRNQ65 24905288 IC50 = 164 nM T80276 COD7I5 24905289 IC50 = 750 nM T80276 C4LP7E 24905290 IC50 = 640 nM T80276 CE9JC2 24905291 IC50 = 403 nM T80276 C2GI1R 24905292 IC50 = 3500 nM T80276 CHW8C4 24905293 IC50 = 276 nM T80276 CQF0H1 24905294 IC50 = 68 nM T80276 CNO7X0 24905295 IC50 = 135 nM T80276 C5WRG7 24905296 IC50 = 135 nM T80276 CQ1S0U 24905297 IC50 = 1900 nM T80276 C4UES7 24905298 IC50 = 615 nM T80276 CMS69P 24905299 IC50 = 100000 nM T80276 CC0U5M 24905300 IC50 = 225 nM T80276 CW7X6S 24905301 IC50 = 5250 nM T80276 C97IQV 24905302 IC50 = 525 nM T80276 CSJ47V 24905303 IC50 = 2660 nM T80276 CPN74C 24905304 IC50 = 6290 nM T80276 C5CS3N 24905305 IC50 = 3850 nM T80276 CK4XE9 24905307 IC50 = 1099 nM T80276 CTU6Z3 24905308 IC50 = 100000 nM T80276 C9SQX1 24905309 IC50 = 5760 nM T80276 CM75JP 24905310 IC50 = 9150 nM T80276 C9Q2BJ 24905311 IC50 = 2260 nM T80276 C9VUA1 24905312 IC50 = 863 nM T80276 CU3RS1 24905313 IC50 = 2220 nM T80276 CYG3H2 24905314 IC50 = 1630 nM T80276 CV5Q7O 24905315 IC50 = 347 nM T80276 C8SA3O 24905316 IC50 = 192 nM T80276 CI5MN3 24905317 IC50 = 113 nM T80276 CJ1P7K 24905318 IC50 = 293 nM T80276 C1T6YQ 24905319 IC50 = 650 nM T80276 CAU86X 24905320 IC50 = 660 nM T80276 C54ISY 24905321 IC50 = 6520 nM T80276 C2GE5I 24905322 IC50 = 1620 nM T80276 C8D6YK 24905323 IC50 = 4870 nM T80276 C5NZH9 24905324 IC50 = 784 nM T80276 C9D6JR 24905325 IC50 = 482 nM T80276 CLZT41 24905326 IC50 = 176 nM T80276 CW8FD3 24905327 IC50 = 244 nM T80276 CHB7A2 24905328 IC50 = 693 nM T80276 CA8EI3 24905329 IC50 = 394 nM T80276 CCQ0O7 24905330 IC50 = 464 nM T80276 CJ81AS 24905331 IC50 = 70 nM T80276 C8PW4H 24905332 IC50 = 76 nM T80276 C2Y5TF 24905333 IC50 = 142 nM T80276 CH9FL5 24905334 IC50 = 1500 nM T80276 C1S0PC 24905335 IC50 = 570 nM T80276 C8N9MV 24905336 IC50 = 1700 nM T80276 C9E8BJ 24905338 IC50 = 2500 nM T80276 CX85AC 24905341 IC50 = 12900 nM T80276 CKZ80E 24905342 IC50 = 175 nM T80276 CO8SH1 24905343 IC50 = 80 nM T80276 C7IZL6 24905344 IC50 = 3100 nM T80276 C3IYB2 24936050 IC50 = 6 nM T80276 CLD3X6 24936051 IC50 = 11 nM T80276 C43VSW 24936353 IC50 = 630.96 nM T80276 C98MEW 24946175 IC50 = 4.8 nM T80276 CC7H3U 24946706 IC50 = 1.1 nM T80276 CDWQ10 24947414 Ki = 2 nM T80276 C78NJE 24955795 IC50 = 2847 nM T80276 C8P6NT 24956158 IC50 = 2666 nM T80276 CJI29P 24956159 IC50 = 11330 nM T80276 CD5HQ0 24969301 IC50 > 10000 nM T80276 CEN9U4 24970086 IC50 = 29 nM T80276 CCZO17 24970164 IC50 = 22 nM T80276 CXI65T 24983588 IC50 > 30000 nM T80276 CH6Q7Y 24983749 IC50 > 30000 nM T80276 C6Q8HD 24983903 IC50 = 2600 nM T80276 C7NYZ4 24984057 IC50 > 30000 nM T80276 CV79PK 24984058 IC50 = 20100 nM T80276 CX24TD 24985362 IC50 > 30000 nM T80276 CV5OB6 24985365 IC50 = 12600 nM T80276 C8QPN6 24992904 IC50 = 3 nM T80276 C6C4RH 24993871 IC50 = 21 nM T80276 CS3Q8B 24995659 Ki > 4000 nM T80276 CGSE92 25009673 Ki = 41 nM T80276 CB5M0S 25023739 IC50 = 6 nM T80276 C0XGE2 25023740 IC50 = 21 nM T80276 CC9OD2 25023741 IC50 = 3 nM T80276 CW14CK 25023742 IC50 = 4 nM T80276 CWHR07 25023743 IC50 = 36 nM T80276 C0JT9A 25023744 IC50 = 2450 nM T80276 CEW91Q 25032963 IC50 = 24 nM T80276 CY50OT 25052783 IC50 = 295 nM T80276 CHR51O 25057242 IC50 = 95 nM T80276 CTM16Y 25069911 IC50 = 4379 nM T80276 CVI2S5 25070227 IC50 = 3477 nM T80276 CNL4Y2 25070228 IC50 = 3787 nM T80276 CSDN18 25070229 IC50 = 3902 nM T80276 CK92QL 25070230 IC50 = 3769 nM T80276 CKZ7X2 25070231 IC50 = 1760 nM T80276 C0T4NK 25070551 IC50 = 57 nM T80276 C1UKQ4 25070552 IC50 = 189 nM T80276 CZRA03 25070553 IC50 = 199 nM T80276 CO20FT 25070554 IC50 = 75 nM T80276 CL4B5Z 25070555 IC50 = 248 nM T80276 C7U0SC 25070882 IC50 = 45 nM T80276 CCN36H 25071204 IC50 = 14 nM T80276 CQ7P4X 25071206 IC50 = 16 nM T80276 C14SFA 25071208 IC50 = 42 nM T80276 CNCJ40 25071516 IC50 = 94 nM T80276 CXWO13 25071518 IC50 = 65 nM T80276 CBH13R 25071519 IC50 = 42 nM T80276 CJM7O0 25071520 IC50 = 70 nM T80276 C68PFD 25073081 IC50 = 66 nM T80276 CBJ20X 25073385 IC50 = 55 nM T80276 CZN7W0 25073388 IC50 = 40 nM T80276 CD69RK 25097993 IC50 = 1300 nM T80276 C8DG4R 25109014 IC50 = 7 nM T80276 CB3W1F 25109202 IC50 = 8.5 nM T80276 CTO19H 25109378 IC50 = 1 nM T80276 C83WVR 25109494 IC50 = 3 nM T80276 CIB90Z 25109643 IC50 = 9 nM T80276 CV1N4E 25109782 Ki = 2 nM T80276 CLP07J 25110819 IC50 > 10000 nM T80276 CK2IJ4 25121551 IC50 = 9 nM T80276 CVM89J 25128663 IC50 = 3981.07 nM T80276 C4HRL9 25128667 IC50 = 316.23 nM T80276 C4SWT5 25128668 IC50 > 79432.82 nM T80276 CIO6A4 25129024 IC50 > 50118.72 nM T80276 CLS7P0 25129381 IC50 = 12589.25 nM T80276 C9R2EA 25129383 IC50 > 100000 nM T80276 C4YZL9 25129386 IC50 = 5011.87 nM T80276 CDO9Q0 25129729 IC50 > 15848.93 nM T80276 CX86YV 25129734 IC50 = 199.53 nM T80276 CA2K4U 25130429 IC50 > 100000 nM T80276 C1J8KH 25132804 IC50 > 50118.72 nM T80276 CI04XW 25132806 IC50 = 25118.86 nM T80276 C5WC4L 25133141 IC50 = 15848.93 nM T80276 CSH37X 25133142 IC50 > 3981.07 nM T80276 CW3HN6 25133144 IC50 = 1584.89 nM T80276 C2CXH3 25165371 IC50 > 10000 nM T80276 CQWL59 25165372 IC50 > 10000 nM T80276 CL87JW 25165773 IC50 = 6000 nM T80276 CB89TL 25165774 IC50 > 10000 nM T80276 CFZI92 25165961 IC50 = 4700 nM T80276 CK2YI4 25168990 IC50 = 912.01 nM T80276 CU4ZH9 25169523 IC50 = 4000 nM T80276 C7G1ZM 25169579 IC50 = 630 nM T80276 CL81FJ 25169580 IC50 = 740 nM T80276 C8WL0Z 25169784 IC50 = 150 nM T80276 CLR8M2 25169786 IC50 = 360 nM T80276 CL3UK2 25170000 IC50 = 530 nM T80276 C6WCR7 25170003 IC50 = 4.7 nM T80276 C5PTZ0 25170410 IC50 = 140 nM T80276 CLJR80 25171641 IC50 = 960 nM T80276 C7ZQC2 25171642 IC50 = 110 nM T80276 C7AHP4 25171644 IC50 = 190 nM T80276 CX6BL8 25171852 IC50 = 620 nM T80276 C7TL2N 25171853 IC50 = 2600 nM T80276 C6BR3F 25171855 IC50 = 2.9 nM T80276 CMI85O 25171856 IC50 = 3.8 nM T80276 CUN9F3 25171857 IC50 = 16 nM T80276 CKY81J 25172061 IC50 = 130 nM T80276 CC1D8V 25172062 IC50 = 0.5 nM T80276 C1L6GX 25172063 IC50 = 36 nM T80276 CFO08N 25172065 IC50 = 21 nM T80276 C8ZF0A 25172066 IC50 = 700 nM T80276 CCW80B 25172270 IC50 = 65 nM T80276 C9HUB6 25172271 IC50 = 55 nM T80276 CC60ZY 25172272 IC50 = 13 nM T80276 C54EGX 25172274 IC50 = 990 nM T80276 C5QVC7 25172275 IC50 = 350 nM T80276 CPW2D9 25172477 IC50 = 0.8 nM T80276 CVDC60 25172479 IC50 = 13 nM T80276 CI6W9H 25172661 IC50 = 0.5 nM T80276 CL5IC0 25172662 IC50 = 82 nM T80276 CDAO95 25172663 IC50 = 77 nM T80276 C8JC3P 25172664 IC50 = 17 nM T80276 CK38ER 25172665 IC50 = 11 nM T80276 C3JI1Y 25172666 IC50 = 40 nM T80276 CXG59Q 25175568 IC50 = 22950 nM T80276 C1C9ZF 25182020 Ki = 113 nM T80276 CUA41N 25182022 Ki = 105 nM T80276 CX2N5M 25182023 Ki = 32 nM T80276 CV6EU9 25182024 Ki = 333 nM T80276 C46ZAW 25182142 Ki = 148 nM T80276 C06EGS 25182144 Ki = 1550 nM T80276 CP17FV 25182145 Ki = 61 nM T80276 CGQ56K 25182146 Ki = 605 nM T80276 C9G6DH 25182281 Ki = 18 nM T80276 CS07FL 25182282 Ki = 128 nM T80276 C2LYI1 25182285 Ki = 47 nM T80276 C7GAR5 25182286 Ki = 40 nM T80276 C9X3OT 25182424 Ki = 46 nM T80276 C0JBX1 25182427 Ki = 44 nM T80276 CAG4R1 25182562 Ki = 144 nM T80276 C5JD1M 25182565 Ki = 102 nM T80276 CWIH67 25182709 Ki = 31 nM T80276 C6O1VG 25182710 Ki = 53 nM T80276 C80UYN 25182711 Ki = 59 nM T80276 C8H9ET 25182714 Ki = 141 nM T80276 CD8M0G 25182867 Ki = 58 nM T80276 C9T6AZ 25182868 Ki = 48 nM T80276 C0S4YF 25182871 Ki = 114 nM T80276 CS4N6U 25183031 Ki = 53 nM T80276 CX8F3W 25183032 Ki = 85 nM T80276 C38MPQ 25195571 IC50 = 270 nM T80276 C1CL7V 25195572 IC50 = 16.5 nM T80276 CD4L2F 25195682 IC50 = 55 nM T80276 C4QTX9 25195788 IC50 = 86 nM T80276 CIRE40 25195789 IC50 = 401 nM T80276 CHJM38 25195893 IC50 = 29 nM T80276 C64SIJ 25195997 IC50 = 708 nM T80276 CB6CP3 25196219 IC50 = 317 nM T80276 CWN52I 25196221 IC50 = 234 nM T80276 C8RWY2 25196900 IC50 = 6000 nM T80276 CNU28R 25197239 IC50 = 83 nM T80276 CMST49 25197240 IC50 = 257 nM T80276 CLW96O 25207689 IC50 = 4 nM T80276 CRO09K 25211064 IC50 > 10000 nM T80276 C6MR3O 25229450 IC50 = 801 nM T80276 CQL23A 25229526 IC50 = 1962 nM T80276 CWP29U 25242324 IC50 = 3.4 nM T80276 CARX27 25253230 IC50 = 3 nM T80276 C58WEU 25260757 IC50 = 1180 nM T80276 C9V5KO 25260758 IC50 = 1301 nM T80276 C8RYX7 25260759 IC50 = 227 nM T80276 C47RYE 25260913 IC50 = 2021 nM T80276 C96OGS 25260915 IC50 = 41 nM T80276 CBCF51 25261227 IC50 = 1616 nM T80276 C5DQF0 25261230 IC50 = 345 nM T80276 C4V2EJ 25261231 IC50 = 100 nM T80276 C3I9SN 25261388 IC50 = 2746 nM T80276 C7SNP6 25261389 IC50 = 1803 nM T80276 C4R3ZS 25261390 IC50 = 1475 nM T80276 CUR93V 25261554 IC50 = 4320 nM T80276 CCR83Z 25261555 IC50 = 613 nM T80276 C38UOX 25262174 IC50 = 677 nM T80276 CD27XK 25262616 IC50 = 270 nM T80276 CPLM23 25262617 IC50 = 1249 nM T80276 CU6C8J 25262782 IC50 = 66 nM T80276 CT97DF 25262783 IC50 = 148 nM T80276 CFL6G2 25262946 IC50 = 247 nM T80276 C3IDN0 25266674 IC50 = 31622.78 nM T80276 CU09IM 26699441 IC50 = 61000 nM T80276 CBY15M 33845371 EC50 = 17800 nM T80276 C2IM0O 39733146 IC50 = 7943.28 nM T80276 CO4PL8 42606076 IC50 = 5120 nM T80276 C20VGT 42606077 IC50 = 360 nM T80276 C7N5EC 42606078 IC50 = 1050 nM T80276 CI69YO 42606079 IC50 > 100000 nM T80276 C5L7IT 42606080 IC50 = 1850 nM T80276 CG04LZ 42606083 IC50 > 100000 nM T80276 C0WEU1 42606190 IC50 > 100000 nM T80276 CD6LN3 42606191 IC50 > 100000 nM T80276 CWR7P5 42606194 IC50 > 100000 nM T80276 CJ2GM1 42606195 IC50 > 100000 nM T80276 C61JUL 42606196 IC50 > 100000 nM T80276 C9GS8P 42606431 IC50 = 3050 nM T80276 CIF63E 42623219 IC50 = 10000 nM T80276 C3DNM9 42623223 IC50 = 2511.89 nM T80276 COR5I0 42623224 IC50 > 19952.62 nM T80276 CX1DC2 42623385 IC50 = 158.49 nM T80276 CR6N3I 42623632 IC50 = 3162.28 nM T80276 C4EM0W 42623869 IC50 = 2511.89 nM T80276 C5TY9Q 42623950 IC50 > 15848.93 nM T80276 CG8Q0C 42630822 IC50 = 22 nM T80276 CYJK74 42632991 IC50 = 354 nM T80276 CQW60S 42632992 IC50 = 178 nM T80276 C2FIY7 42633175 IC50 = 340 nM T80276 CL2XD7 42633904 IC50 = 1996 nM T80276 C9B0DZ 42633906 IC50 = 4207 nM T80276 CHP49D 42635321 IC50 = 70 nM T80276 C96ETP 42635322 IC50 = 65 nM T80276 CZN3G1 42635323 IC50 = 1506 nM T80276 CCV0R1 42635502 IC50 = 7500 nM T80276 CR8C3W 42635504 IC50 = 21 nM T80276 C10RBA 42636535 IC50 = 15 nM T80276 CY07TS 43845722 IC50 = 370 nM T80276 C3ROX1 44124863 Ki = 1.4 nM T80276 C2YQX8 44125256 Ki = 11 nM T80276 CV5O8L 44125375 Ki = 3.3 nM T80276 C5JN4O 44125376 Ki = 2.8 nM T80276 C0U2OY 44125377 Ki = 1.2 nM T80276 CI3K7H 44129042 IC50 = 71 nM T80276 CIE0J3 44129043 IC50 = 84 nM T80276 CUW85V 44129044 IC50 = 24 nM T80276 C2B9DE 44129118 IC50 = 39 nM T80276 C6O0JA 44129197 IC50 = 30 nM T80276 C0R1PH 44129198 IC50 = 550 nM T80276 C6LGD5 44129200 IC50 = 44 nM T80276 C03RLS 44129270 IC50 = 520 nM T80276 CTG8U7 44129271 IC50 = 14 nM T80276 CDQ56T 44129272 IC50 = 1200 nM T80276 CU4H1I 44129274 IC50 = 39 nM T80276 C79QOC 44129275 IC50 = 33 nM T80276 C0W3ZF 44129348 IC50 = 170 nM T80276 CQ5UJ4 44129350 IC50 = 100 nM T80276 CH6RO4 44129351 IC50 = 180 nM T80276 CPAU59 44129353 IC50 = 88 nM T80276 CN5O4I 44129429 IC50 = 26 nM T80276 CON25C 44129430 IC50 = 160 nM T80276 C3ZSV2 44129432 IC50 = 70 nM T80276 C3MWZ1 44129511 IC50 = 20 nM T80276 CM5U2I 44137407 IC50 = 95 nM T80276 CQ82MS 44138035 IC50 = 7000 nM T80276 C5CQK3 44138092 IC50 = 66 nM T80276 CZA3N9 44138128 IC50 = 5000 nM T80276 CP61GU 44156032 IC50 = 59 nM T80276 C3CBU7 44156033 IC50 = 1013 nM T80276 C7XI2W 44156156 IC50 = 200 nM T80276 C63BLR 44156157 IC50 = 2300 nM T80276 C19LGE 44158465 IC50 = 25 nM T80276 CG4DY5 44158569 IC50 = 53 nM T80276 CB46RQ 44159380 IC50 = 89 nM T80276 CO9RT8 44180017 IC50 = 16 nM T80276 CF17OS 44180029 IC50 = 551 nM T80276 CHK8Z6 44180034 IC50 = 714 nM T80276 CEJ5F7 44180035 IC50 = 110 nM T80276 CQNT23 44180155 IC50 = 1857 nM T80276 CIKM57 44180156 IC50 = 34 nM T80276 CBP2T3 44180157 IC50 = 72 nM T80276 CHB2D9 44180158 IC50 = 14 nM T80276 CC9LU0 44180268 IC50 = 1.4 nM T80276 C9CGB4 44180282 IC50 = 242 nM T80276 C2S5LC 44180395 IC50 = 56 nM T80276 C40NOQ 44180397 IC50 = 345 nM T80276 CTB46H 44180398 IC50 = 400 nM T80276 COT92S 44180509 IC50 = 24000 nM T80276 C10TLO 44180511 IC50 = 14000 nM T80276 CXO26U 44180615 IC50 = 8.3 nM T80276 CE30IL 44180626 IC50 = 53 nM T80276 C93MZI 44180629 IC50 = 109 nM T80276 CL2TK9 44180738 IC50 = 187 nM T80276 CGCR01 44180740 IC50 = 86 nM T80276 CXV78M 44180743 IC50 = 71 nM T80276 CAS3X6 44180851 IC50 = 66 nM T80276 CRS2G3 44180853 IC50 = 1006 nM T80276 CSTZ70 44181062 IC50 = 1.4 nM T80276 C9HU7V 44181276 IC50 = 80 nM T80276 CBW86O 44181374 IC50 = 3 nM T80276 CK3A7D 44181481 IC50 = 4.9 nM T80276 C2VZX7 44181492 IC50 = 176 nM T80276 C7SYM2 44181493 IC50 = 294 nM T80276 CB8KF1 44181494 IC50 = 682 nM T80276 C5AI8R 44181598 IC50 = 556 nM T80276 CK03RW 44181599 IC50 = 4598 nM T80276 CXL61J 44181600 IC50 = 297 nM T80276 C6TZK5 44181601 IC50 = 75 nM T80276 CCIV74 44181602 IC50 = 61 nM T80276 C36WUP 44181603 IC50 = 7158 nM T80276 CS2U7R 44181604 IC50 = 154 nM T80276 CL6W0C 44181605 IC50 = 77 nM T80276 CA6QG9 44181707 IC50 = 1.4 nM T80276 C9G2LH 44181709 IC50 = 29 nM T80276 CFD41Z 44181718 IC50 = 4539 nM T80276 C2RB1P 44181719 IC50 = 699 nM T80276 CMC75I 44181720 IC50 = 238 nM T80276 CWTS93 44181721 IC50 = 116 nM T80276 CT1JL2 44181722 IC50 = 112 nM T80276 CE9HO1 44181723 IC50 = 100 nM T80276 CFSB29 44181724 IC50 = 217 nM T80276 CO0YZ7 44182308 IC50 = 548 nM T80276 CS0M9A 44187604 IC50 = 5 nM T80276 C0BRI9 44187779 IC50 = 8 nM T80276 CDA81B 44187783 IC50 = 9.5 nM T80276 C0LB8S 44187784 IC50 = 2.5 nM T80276 CCTO21 44187951 IC50 = 23.3 nM T80276 CVYS60 44187952 IC50 = 1 nM T80276 C8X3UZ 44187955 IC50 = 2.4 nM T80276 CJU85Z 44188321 IC50 = 6 nM T80276 CHU02A 44188322 IC50 = 3 nM T80276 C69HQS 44188840 IC50 = 6 nM T80276 CD78AG 44188841 IC50 = 3 nM T80276 CY7EL1 44188842 IC50 = 5 nM T80276 C0SE1X 44188843 IC50 = 10.5 nM T80276 CG13ZF 44188844 IC50 = 3.5 nM T80276 CR0BF9 44189010 IC50 = 25 nM T80276 C71NFL 44189011 IC50 = 23.5 nM T80276 C39ABJ 44189192 IC50 = 3.6 nM T80276 CK73NR 44219749 IC50 = 1026 nM T80276 C2V6WY 44232672 IC50 = 47 nM T80276 CA91IW 44232914 IC50 = 404 nM T80276 CN10TK 44232915 IC50 = 2005 nM T80276 CNY95J 44232916 IC50 = 631 nM T80276 COXT27 44232917 IC50 = 284 nM T80276 CFC2A1 44232918 IC50 = 23 nM T80276 CVN7P2 44233160 IC50 = 14 nM T80276 CQXD21 44233161 IC50 = 211 nM T80276 CI7N6F 44233162 IC50 = 225 nM T80276 CC6H5K 44233163 IC50 = 149 nM T80276 CSGQ48 44233164 IC50 = 209 nM T80276 CI65AN 44233388 IC50 = 681 nM T80276 CS9UA8 44233389 IC50 = 490 nM T80276 CZ3L7W 44233390 IC50 = 505 nM T80276 CA7R1U 44233391 IC50 = 661 nM T80276 CN4A7W 44233639 IC50 = 35 nM T80276 CWLA98 44233640 IC50 = 18 nM T80276 CXO1L7 44233641 IC50 = 15 nM T80276 C96DJK 44241762 Ki = 23 nM T80276 C92UIQ 44241764 Ki = 30 nM T80276 C8XCS6 44242164 Ki = 1 nM T80276 CFC1E3 44242168 Ki = 3 nM T80276 C1EDX6 44242233 IC50 < 1.4 nM T80276 CY0C8Q 44242297 IC50 = 12 nM T80276 CN1BK0 44242299 Ki = 0.6 nM T80276 C5YT6K 44242362 Ki = 1.2 nM T80276 CJ27VR 44242423 Ki = 11 nM T80276 COW73L 44242425 Ki = 31 nM T80276 CG9DF3 44242426 Ki = 1.5 nM T80276 CT6AD8 44242428 Ki = 1 nM T80276 C0RO4N 44242493 IC50 = 52 nM T80276 CM1Z7F 44242776 Ki = 5 nM T80276 CJ8QI0 44242777 Ki = 4 nM T80276 CU2F9E 44413107 IC50 = 340 nM T80276 C9SK8P 44413114 IC50 = 600 nM T80276 C9DT8F 44426432 IC50 = 560 nM T80276 CS17AZ 44426433 IC50 > 30000 nM T80276 C59FBV 44426434 IC50 = 1700 nM T80276 CUY2J9 44426435 IC50 = 160 nM T80276 CC65DT 44426437 IC50 = 2400 nM T80276 C6SPI8 44426438 IC50 > 30000 nM T80276 CFA7N5 44426448 IC50 = 100 nM T80276 CQN40C 44426456 IC50 = 24 nM T80276 C98MAL 44436951 IC50 = 860 nM T80276 CD0ME6 44436952 IC50 > 10000 nM T80276 CR6ZU9 44436953 IC50 > 10000 nM T80276 CYK0T1 44436954 IC50 > 10000 nM T80276 CYV15O 44436955 IC50 > 10000 nM T80276 C3M4RN 44436961 IC50 > 10000 nM T80276 CA4SV2 44436964 IC50 = 5000 nM T80276 CO5FK1 44436967 IC50 > 10000 nM T80276 CRKU98 44436970 IC50 > 10000 nM T80276 C9V1SZ 44436971 IC50 > 10000 nM T80276 CZ4V2L 44436972 IC50 = 2300 nM T80276 COG34Q 44436976 IC50 > 10000 nM T80276 C4RAK8 44436979 IC50 = 2200 nM T80276 CXN93Q 44436980 IC50 > 10000 nM T80276 CX57RI 44436981 IC50 > 10000 nM T80276 C9ZML1 44454396 IC50 = 56 nM T80276 C2QF1N 44457157 IC50 = 90 nM T80276 C34HLQ 44457158 IC50 = 56 nM T80276 CSW53V 44457165 IC50 = 91 nM T80276 CZ4O2K 44457166 IC50 = 43 nM T80276 C6JS1G 44457167 IC50 = 87 nM T80276 CW5KH3 44457168 IC50 = 199 nM T80276 CCBP46 44457169 IC50 = 444 nM T80276 CWTU20 44457172 IC50 = 918 nM T80276 C2QR9D 44457173 IC50 = 193 nM T80276 C9H2FA 44457174 IC50 = 1580 nM T80276 C9X8CD 44457178 IC50 = 127 nM T80276 CD4RP9 44457179 IC50 = 15 nM T80276 C16ASL 44457183 IC50 = 22 nM T80276 CA04RG 44457184 IC50 = 10 nM T80276 C8INQ7 44457185 IC50 = 24 nM T80276 C0UBI8 44457188 IC50 = 50 nM T80276 CGCS67 44457189 IC50 = 24 nM T80276 C9WG2B 44457191 IC50 = 12 nM T80276 C4OK8P 44457192 IC50 = 5 nM T80276 CHSE37 44457195 IC50 = 8.4 nM T80276 CN9H7F 44457201 IC50 = 104 nM T80276 CI6G5C 44457211 IC50 = 60 nM T80276 C9N4PA 44457212 IC50 = 37 nM T80276 CB70NU 44457213 IC50 = 9.6 nM T80276 CY4H8C 44457218 IC50 = 63 nM T80276 C0RN9S 44457220 IC50 = 33 nM T80276 C2JV8Y 44457231 IC50 = 172 nM T80276 CQD4T3 44457232 IC50 = 31 nM T80276 CT02VO 44457235 IC50 = 38 nM T80276 CB2J6E 44457236 IC50 = 78 nM T80276 CG7YT9 44457237 IC50 = 45 nM T80276 CVG75D 44473371 IC50 = 0.4 nM T80276 C30NZA 44475985 IC50 = 34 nM T80276 CAT8F7 44475986 IC50 = 788 nM T80276 CSR73H 44475987 IC50 = 85000 nM T80276 CDAX92 44475988 IC50 = 53 nM T80276 CBH0S5 44475989 IC50 = 3438 nM T80276 CW5A7L 44475990 IC50 = 137 nM T80276 CLKU13 44481151 IC50 = 110 nM T80276 CX3FK1 44513884 IC50 = 3 nM T80276 CL4RO5 44513885 IC50 = 1.7 nM T80276 C6RC9J 44513886 IC50 = 3 nM T80276 CGS7Q4 44513887 IC50 = 2 nM T80276 CSVD32 44513888 IC50 = 16.5 nM T80276 CLN2M5 44514201 IC50 = 6.5 nM T80276 C2Y8ML 44514203 IC50 = 19.5 nM T80276 CA9H8D 44514205 IC50 = 60.5 nM T80276 C01ZJI 44514208 IC50 = 1 nM T80276 CZ8WK6 44514210 IC50 = 3 nM T80276 CI8H3K 44514481 IC50 = 247.5 nM T80276 C51SEJ 44515083 IC50 = 1.5 nM T80276 CXBV98 44515084 IC50 = 1 nM T80276 C73HNB 44515696 IC50 = 12.5 nM T80276 CB7XW5 44516307 IC50 = 6 nM T80276 C4W5EM 44516309 IC50 = 0.5 nM T80276 C8VAU1 44516310 IC50 = 1.5 nM T80276 C8I1ZB 44516311 IC50 = 0.4 nM T80276 CSJ95V 44516635 IC50 = 0.7 nM T80276 CV6Z0N 44516636 IC50 = 0.6 nM T80276 CB3MV8 44517288 IC50 = 3 nM T80276 CDEQ97 44520808 IC50 = 36 nM T80276 CT7DW6 44520809 IC50 = 69 nM T80276 C3T2YD 44520810 IC50 = 50 nM T80276 CJP71L 44520811 IC50 = 86 nM T80276 CB4RN0 44520812 IC50 = 31 nM T80276 CGQ1F8 44520814 IC50 = 244 nM T80276 C2W5QS 44520815 IC50 = 2766 nM T80276 CN78XU 44520816 IC50 = 466 nM T80276 C1TI9F 44520817 IC50 = 4394 nM T80276 CHS6C1 44520818 IC50 = 1112 nM T80276 CKP60Q 44520819 IC50 = 238 nM T80276 C0XEA9 44520820 IC50 = 1008 nM T80276 CFE63J 44520821 IC50 = 1272 nM T80276 CV43BN 44520822 IC50 = 520 nM T80276 CYU2B5 44520824 IC50 = 1310 nM T80276 C73ZYA 44520825 IC50 = 5870 nM T80276 CB25DI 44539683 IC50 = 63 nM T80276 CNWO35 44539684 IC50 = 30 nM T80276 C8MTO3 44539685 IC50 = 249 nM T80276 CTQ06N 44539783 IC50 = 128 nM T80276 C03IGD 44540030 IC50 = 25118.86 nM T80276 C5LWU1 44540126 IC50 = 19952.62 nM T80276 CYD4Z8 44540130 IC50 = 316.23 nM T80276 CAT2R7 44540316 IC50 = 25118.86 nM T80276 C2T9GC 44540407 IC50 = 10000 nM T80276 CQ4PE7 44540492 IC50 > 25118.86 nM T80276 C3D8CF 44540543 IC50 = 63 nM T80276 C0Z3QI 44540642 IC50 = 233 nM T80276 C3Z7GL 44540644 IC50 = 43 nM T80276 CGB2A8 44540925 IC50 = 580 nM T80276 CFI4O2 44541101 IC50 > 10000 nM T80276 CG9DO4 44543764 Ki = 10 nM T80276 CW19QS 44544943 Ki = 3 nM T80276 C6L4SV 44545041 Ki = 2 nM T80276 C0IX1C 44545849 IC50 = 2 nM T80276 C6HC3L 44548482 IC50 = 3.2 nM T80276 CH3L9P 44551660 IC50 = 1490 nM T80276 CYMD49 44552663 IC50 = 37 nM T80276 C6B7LH 44552664 IC50 = 5 nM T80276 C3QZX0 44552666 IC50 = 9 nM T80276 C64OQC 44552667 IC50 = 11 nM T80276 C7LG6Q 44552844 IC50 = 5 nM T80276 C9T2CZ 44552845 IC50 = 8 nM T80276 CXLD75 44552846 IC50 = 6 nM T80276 CALT95 44554240 IC50 = 1034 nM T80276 CVDA08 44554755 IC50 = 542 nM T80276 C25EGX 44554909 IC50 = 800 nM T80276 C6VR1P 44554910 IC50 = 1580 nM T80276 CR4J0X 44554913 IC50 = 422 nM T80276 CWV2T9 44554915 IC50 = 15 nM T80276 CCW12H 44555222 IC50 = 30 nM T80276 CTM8S9 44555225 IC50 = 40 nM T80276 C7PSO6 44555226 IC50 = 42 nM T80276 C3VRO9 44557921 IC50 = 2454.71 nM T80276 CRE61W 44577592 IC50 = 677 nM T80276 CH63GM 44577593 IC50 = 172 nM T80276 CA8MV5 44577594 IC50 = 1108 nM T80276 C9IXW8 44577638 IC50 = 825 nM T80276 C8A5RT 44577639 IC50 = 116 nM T80276 CNP02V 44577640 IC50 = 164 nM T80276 CT6GN5 44577641 IC50 = 791 nM T80276 C1QN3F 44577827 IC50 = 24.2 nM T80276 C3MGZ9 44577915 IC50 > 20000 nM T80276 CTR89C 44577918 IC50 > 20000 nM T80276 CO05YG 44577919 IC50 = 736 nM T80276 CT70WA 44577920 IC50 = 188 nM T80276 C5KXS4 44577921 IC50 = 917 nM T80276 CZ2HI5 44577922 IC50 = 636 nM T80276 CGTU34 44577950 IC50 = 2900 nM T80276 CQC50R 44577951 IC50 = 294 nM T80276 C8ZTW2 44577952 IC50 = 1131 nM T80276 CIL93G 44577953 IC50 = 1812 nM T80276 C8NB5H 44578037 IC50 > 40000 nM T80276 CX9TO2 44578038 IC50 = 20280 nM T80276 C7AHR4 44578039 IC50 > 50000 nM T80276 C13LGI 44578040 IC50 > 50000 nM T80276 CNZ06H 44578074 IC50 = 20060 nM T80276 C41TYA 44578108 IC50 = 107 nM T80276 C2W3SQ 44578109 IC50 = 125 nM T80276 C40VHS 44580686 IC50 = 243 nM T80276 CT0R7C 44581248 IC50 = 0.8 nM T80276 CL8S0Y 44592136 IC50 >= 50000 nM T80276 C9E6JV 44592170 IC50 >= 10000 nM T80276 C8DUA1 44592171 IC50 > 10000 nM T80276 CGP6M7 44592216 IC50 = 20000 nM T80276 CS38JL 44592217 IC50 = 100000 nM T80276 CJ1FW0 44592218 IC50 > 100000 nM T80276 CVB1I3 44592259 IC50 > 100000 nM T80276 CV9MY8 44592260 IC50 > 100000 nM T80276 CA65CE 44592261 IC50 = 100000 nM T80276 CEHY48 44592262 IC50 > 100000 nM T80276 C09OLK 44592299 IC50 = 29000 nM T80276 CJM35R 44592300 IC50 > 100000 nM T80276 C54DKW 44592302 IC50 = 100000 nM T80276 CJX76V 44592338 IC50 > 100000 nM T80276 CNY53M 44592339 IC50 > 100000 nM T80276 CXPK04 44592340 IC50 > 100000 nM T80276 C0L2HO 44593630 IC50 = 738 nM T80276 C2NQ6Z 44593631 IC50 = 89 nM T80276 CY3SV7 44596118 IC50 = 3900 nM T80276 C5VNA7 44599029 IC50 = 5 nM T80276 CCFX21 44599203 IC50 = 10 nM T80276 CU5YK1 44599206 IC50 = 6 nM T80276 C4OP3Y 44599690 IC50 = 0.9 nM T80276 C7H0XM 44599855 IC50 = 2.4 nM T80276 CL73YV 44600010 IC50 = 1.8 nM T80276 C54ZQB 44600166 IC50 = 0.8 nM T80276 C2ZYD0 44600649 IC50 = 1.4 nM T80276 C3R2PX 44600650 IC50 = 80 nM T80276 C8AT9I 44600651 IC50 = 43 nM T80276 C5JL6C 44600806 IC50 = 28 nM T80276 CJUQ51 44600808 IC50 = 76 nM T80276 C0BXS4 44600809 IC50 = 42 nM T80276 CA9LP4 44600952 IC50 = 16 nM T80276 CFK83C 44600954 IC50 = 142 nM T80276 CX30VY 44600955 IC50 = 8 nM T80276 C9N1SY 44600956 IC50 = 24 nM T80276 CUI9Y8 44601112 IC50 = 226 nM T80276 CBV38N 44601113 IC50 = 54 nM T80276 CA3K8E 44601278 IC50 = 30 nM T80276 CZX94G 44601279 IC50 = 53 nM T80276 CD1A2Z 44601448 IC50 = 36 nM T80276 CB12CS 44601449 IC50 = 42 nM T80276 CIDT64 44601450 IC50 = 7 nM T80276 CWY15L 44604823 IC50 = 323 nM T80276 CN9ZD0 44604824 IC50 = 30 nM T80276 CL3S1F 44604825 IC50 = 1005 nM T80276 C28QLM 44605035 IC50 = 801 nM T80276 C75XHS 44605037 IC50 = 41 nM T80276 CFN95D 44605038 IC50 = 17 nM T80276 CD8Q9Z 44605039 IC50 = 10 nM T80276 CI70YP 44605246 IC50 = 34 nM T80276 C36ZFK 44605247 IC50 = 21 nM T80276 CEK25C 44605248 IC50 = 41 nM T80276 C3F4UX 44605249 IC50 = 189 nM T80276 CQ0FZ7 44605426 IC50 = 1207 nM T80276 CC7G2L 44605427 IC50 = 1782 nM T80276 CDLP04 44605428 IC50 = 80 nM T80276 CSKN09 44605429 IC50 = 786 nM T80276 CA79QG 44605430 IC50 = 898 nM T80276 CM49FO 44605789 IC50 = 268 nM T80276 C3DK5F 44605790 IC50 = 721 nM T80276 C9Z4TY 44605791 IC50 = 81 nM T80276 C9F8JY 44605792 IC50 = 4362 nM T80276 CGT58A 44606131 IC50 = 314 nM T80276 CTO96K 44606133 IC50 = 10 nM T80276 CH7O9Y 44606302 IC50 = 602 nM T80276 C8Y4FE 44606303 IC50 = 18 nM T80276 C4PEO6 44606304 IC50 = 194 nM T80276 CG04KF 44606474 IC50 = 2092 nM T80276 C86RYX 44606475 IC50 = 4632 nM T80276 CNI9G3 44606476 IC50 = 4052 nM T80276 CE90UX 44606477 IC50 = 9500 nM T80276 CQIY50 44606640 IC50 = 1935 nM T80276 C1ML5R 44606641 IC50 = 553 nM T80276 C35QOE 44606642 IC50 = 521 nM T80276 CWQ67K 44606643 IC50 = 4546 nM T80276 CY0QH9 44606644 IC50 = 517 nM T80276 CFQT17 44606818 IC50 = 792 nM T80276 C84TLP 44606820 IC50 = 4058 nM T80276 C3H4EB 44606823 IC50 = 231 nM T80276 CD4A8G 44606998 IC50 = 436 nM T80276 C80RQK 44606999 IC50 = 290 nM T80276 CFW9G3 44607000 IC50 = 59 nM T80276 CHL59X 44607001 IC50 = 1000 nM T80276 C7H3RM 44607002 IC50 = 1050 nM T80276 C2TJ3K 44607003 IC50 = 137 nM T80276 CHM5T4 44607180 IC50 = 493 nM T80276 C85XWN 44607181 IC50 = 1368 nM T80276 C52ILQ 44607183 IC50 = 486 nM T80276 C2UP6C 44607528 IC50 = 589 nM T80276 CH6OY3 44607529 IC50 = 1935 nM T80276 CK5MP7 44608114 Ki = 0.8 nM T80276 C6GU1R 44608115 Ki = 1.4 nM T80276 CMU6V8 44608118 Ki = 1.4 nM T80276 CY6IN1 44608268 Ki = 200 nM T80276 CH27SA 44608430 Ki = 3.3 nM T80276 CLN65Q 44608432 Ki = 0.9 nM T80276 CH6V9F 44608754 Ki = 0.9 nM T80276 C0IY9N 44608757 Ki = 1.2 nM T80276 C3YLE4 44608758 Ki = 5.7 nM T80276 C90ITS 44608915 Ki = 0.6 nM T80276 C90CGU 44609072 Ki = 3.1 nM T80276 CG5J4V 44609075 Ki = 2.1 nM T80276 CZH1P9 44609387 Ki = 0.8 nM T80276 CNDX48 44609388 Ki = 0.8 nM T80276 CCJW12 44609391 Ki = 0.9 nM T80276 C9YWD7 44609543 Ki = 1.9 nM T80276 CD0Y7Z 44609544 Ki = 1.8 nM T80276 CQ3D6M 44609547 Ki = 1 nM T80276 C7W9HT 44609702 Ki = 38 nM T80276 CBYD58 44609854 Ki = 1.3 nM T80276 C4GBH7 44609857 Ki = 375 nM T80276 CK7D0C 44609858 Ki = 5.1 nM T80276 CS25NQ 44610008 Ki = 856 nM T80276 CQG70K 44610162 Ki = 1 nM T80276 C6CAE8 44610163 Ki = 0.6 nM T80276 CL7DS8 44610316 Ki = 0.9 nM T80276 C73BFI 44610482 Ki = 3.1 nM T80276 C93GAZ 44610483 Ki = 0.8 nM T80276 CBOZ09 44610484 Ki = 1 nM T80276 C4TS8G 44610775 IC50 > 10000 nM T80276 CE95RQ 44620964 IC50 = 1.8 nM T80276 CVYJ36 44620965 IC50 = 5.5 nM T80276 CA8BY7 44621440 IC50 = 12589254.12 nM T80276 C5M1FR 44621441 IC50 = 12589254.12 nM T80276 C5LD7E 44621442 IC50 = 7943282.35 nM T80276 CO4GT0 44621447 IC50 = 12589254.12 nM T80276 CUV26H 44621448 IC50 = 7943282.35 nM T80276 CV2MG9 44621449 IC50 = 10000000 nM T80276 C24IYW 44621451 IC50 = 39810717.06 nM T80276 C0F9YW 44621452 IC50 = 10000000 nM T80276 C0GRD8 44621454 IC50 = 19952623.15 nM T80276 C4YHJ0 44621456 IC50 = 15848931.92 nM T80276 C31VBF 44621458 IC50 = 3981071.71 nM T80276 CAE82W 44623107 Ki = 1.4 nM T80276 C54IUP 44818842 IC50 = 83 nM T80276 C16IMZ 44819024 IC50 = 10.5 nM T80276 CN38JF 44819199 IC50 = 10.5 nM T80276 CVW6L8 44819200 IC50 = 6.5 nM T80276 CZ7M6D 44819201 IC50 = 2.4 nM T80276 C7MU8J 44819203 IC50 = 1.4 nM T80276 C8FU0W 44819375 IC50 = 6.8 nM T80276 C4N8CK 44819376 IC50 = 3.2 nM T80276 CYP0M7 45254032 IC50 > 300 nM T80276 CYV72W 45267273 IC50 = 20 nM T80276 C5I1VH 45379222 IC50 = 350 nM T80276 CA4JZ8 45379223 IC50 = 11 nM T80276 C4V5DT 45482916 IC50 = 5554 nM T80276 CAL96M 45482923 IC50 = 1827 nM T80276 C8T6ML 45482926 IC50 = 4271 nM T80276 C5C2YW 45482931 IC50 = 3877 nM T80276 CP45HK 45482935 IC50 = 704 nM T80276 CR93VD 45482947 IC50 = 5333 nM T80276 CDXB49 45482952 IC50 = 1367 nM T80276 CCS97L 45482982 IC50 = 227 nM T80276 CX4TC8 45483330 IC50 = 5190 nM T80276 CV81ML 45487755 IC50 > 10000 nM T80276 CF3TV5 45488020 IC50 = 3125 nM T80276 CPLM59 45488021 IC50 = 836 nM T80276 CIL9W1 45488031 IC50 = 263 nM T80276 C2Q9ID 45488032 IC50 = 21 nM T80276 CA98FY 45488033 IC50 = 320 nM T80276 CH07NQ 45488034 IC50 < 136 nM T80276 CB8DE0 45488052 IC50 = 40 nM T80276 CF3LV9 45488056 IC50 = 235 nM T80276 CCL46I 45488057 IC50 = 196 nM T80276 CP58QK 45488058 IC50 = 68 nM T80276 C9S4MU 45488059 IC50 = 109 nM T80276 C0V7UL 45488060 IC50 = 102 nM T80276 C8YEC5 45488061 IC50 = 175 nM T80276 C6RTH4 45488066 IC50 = 270 nM T80276 CWN8V6 45488069 IC50 = 282 nM T80276 C1YM6P 45488070 IC50 = 2154 nM T80276 CNK52A 45488071 IC50 = 373 nM T80276 CO8T6V 45488077 IC50 = 51 nM T80276 CBAT68 45488078 IC50 = 1436 nM T80276 CZ68MG 45488079 IC50 = 150 nM T80276 CFOH35 45488080 IC50 = 76 nM T80276 CE3Q7D 45488081 IC50 = 207 nM T80276 CI3FZ2 45488082 IC50 = 256 nM T80276 C4OJT8 45494812 IC50 = 28000 nM T80276 CV1U7I 46180604 IC50 = 2 nM T80276 CED2B3 46180606 IC50 = 2900 nM T80276 CJR31W 46180607 IC50 = 430 nM T80276 CDV85O 46180663 IC50 = 240 nM T80276 C1MP9H 46180664 IC50 = 28 nM T80276 C0T9AE 46180665 IC50 = 16 nM T80276 CZGB46 46180666 IC50 = 3.5 nM T80276 C4HFV9 46190734 IC50 = 27 nM T80276 CTZD58 46190735 IC50 = 35 nM T80276 C61ZLI 46190736 IC50 = 300 nM T80276 C6H3GT 46196486 IC50 = 4 nM T80276 CL08DK 46201895 IC50 = 2.7 nM T80276 CAU17V 46202808 IC50 = 12589.25 nM T80276 C3Z6BX 46206784 IC50 = 17 nM T80276 CX8S2G 46215210 IC50 = 1600 nM T80276 CGMS50 46215563 IC50 = 2300 nM T80276 CRBF57 46215564 IC50 = 17700 nM T80276 CO1D6B 46215565 IC50 = 7600 nM T80276 CZ58FY 46215814 IC50 > 10000 nM T80276 CDA3R9 46220225 IC50 = 6.8 nM T80276 CIJ5V9 46224766 IC50 = 23 nM T80276 CIPV59 46224808 IC50 = 44 nM T80276 C4SQY2 46225156 IC50 = 1053 nM T80276 CL89JZ 46225157 IC50 = 1373 nM T80276 CFB7Y4 46225158 IC50 = 28 nM T80276 CRQ5M4 46225259 IC50 = 6700 nM T80276 C65IPQ 46225280 IC50 = 64 nM T80276 C8A7QJ 46225281 IC50 = 37 nM T80276 CPL45H 46225307 IC50 = 1211 nM T80276 CTN8J2 46225308 IC50 = 2915 nM T80276 CU12LG 46227561 IC50 = 1767 nM T80276 CU0T1P 46227563 IC50 > 10000 nM T80276 CK20PN 46227564 IC50 = 8619 nM T80276 C3VB6I 46227571 IC50 = 4372 nM T80276 CS03RK 46227572 IC50 = 119 nM T80276 CO4J6R 46227578 IC50 = 6199 nM T80276 CO14HC 46227579 IC50 = 80 nM T80276 CM1A2S 46227582 IC50 = 322 nM T80276 CT2CH5 46227596 IC50 = 423 nM T80276 CG26LH 46227597 IC50 = 46 nM T80276 CXW1N8 46227599 IC50 = 1262 nM T80276 CO64ZL 46227600 IC50 = 825 nM T80276 CBF0O4 46227603 IC50 = 874 nM T80276 C2Z4WI 46227604 IC50 = 179 nM T80276 C76PKV 46227605 IC50 = 148 nM T80276 C3JK1T 46227606 IC50 = 12 nM T80276 CV9O8I 46227607 IC50 = 86 nM T80276 CW25EH 46227608 IC50 = 8.3 nM T80276 C5FU9E 46227614 IC50 = 399 nM T80276 C59UJH 46227615 IC50 = 324 nM T80276 CS3A9G 46227620 IC50 = 1359 nM T80276 CG29EB 46227625 IC50 = 82 nM T80276 CI9CJ1 46227632 IC50 = 246 nM T80276 CL34IK 46227801 IC50 = 26 nM T80276 C6D2RL 46227820 IC50 = 25 nM T80276 CSIK15 46228569 IC50 = 1521 nM T80276 C18WPC 46232643 IC50 = 234 nM T80276 CF4WB3 46232644 IC50 = 375 nM T80276 C7LKA5 46232645 IC50 = 966 nM T80276 C3ZP0G 46232682 IC50 = 705 nM T80276 CLE2O9 46232721 IC50 = 648 nM T80276 C4IA5M 46232759 IC50 = 305 nM T80276 C64HAE 46232760 IC50 = 4577 nM T80276 CIMH64 46232761 IC50 = 5129 nM T80276 C47ZSV 46232801 IC50 = 12000 nM T80276 CVF7G6 46232802 IC50 = 353 nM T80276 CXP84Y 46232803 IC50 = 220 nM T80276 CT2O8D 46232804 IC50 = 270 nM T80276 C7RF5Y 46239967 IC50 = 10 nM T80276 CL7C2K 46244173 IC50 = 940 nM T80276 C2NH0A 46244259 IC50 = 2700 nM T80276 CVJM38 46244260 IC50 = 1400 nM T80276 C79JGP 46830152 IC50 = 3477 nM T80276 CC62SY 46830153 IC50 = 4040 nM T80276 CU4T7F 46830277 IC50 = 39 nM T80276 C94YRI 46853654 IC50 = 398.11 nM T80276 CZ3WS1 46861592 IC50 = 0.6 nM T80276 C64MLU 46864999 IC50 = 43 nM T80276 CJ79DE 46865000 IC50 = 90 nM T80276 C7H4YM 46865419 IC50 > 10000 nM T80276 CRO8W0 46865423 IC50 = 3 nM T80276 C47VTS 46865424 IC50 = 2 nM T80276 C7Q4OP 46865531 IC50 < 1 nM T80276 C7T4RN 46865885 IC50 = 899 nM T80276 CO3P0J 46866604 IC50 = 148 nM T80276 C0V2QZ 46866605 IC50 = 41 nM T80276 CQ2Y1V 46866705 Ki = 0.13 nM T80276 C63RCG 46870269 IC50 = 794.33 nM T80276 CTQ25M 46871497 IC50 = 1000 nM T80276 CQB16A 46872415 IC50 > 20000 nM T80276 C62NFQ 46883920 IC50 = 24 nM T80276 CKJ2D4 46883989 IC50 = 311 nM T80276 C82RWD 46883990 IC50 > 10000 nM T80276 CE3B7R 46883991 IC50 = 89 nM T80276 CP9JO4 46884017 IC50 = 498 nM T80276 C18KOY 46884018 IC50 = 2080 nM T80276 C9RD8J 46884019 IC50 = 2220 nM T80276 CP3C4Z 46884064 IC50 = 275 nM T80276 C65AQI 46884065 IC50 = 2030 nM T80276 C7NK1H 46884066 IC50 = 308 nM T80276 C3BV5E 46884067 IC50 = 2660 nM T80276 C9LB7I 46884068 IC50 = 1677 nM T80276 CLOR10 46884069 IC50 = 4598 nM T80276 CE70MJ 46884070 IC50 = 909 nM T80276 CIAK59 46884071 IC50 = 600 nM T80276 CO09QJ 46884072 IC50 = 2310 nM T80276 CK95YV 46884073 IC50 = 1030 nM T80276 CUI09D 46884074 IC50 = 1230 nM T80276 CUL4I2 46884075 IC50 = 1570 nM T80276 C9MHF4 46884076 IC50 > 10000 nM T80276 CHM48L 46884077 IC50 = 4960 nM T80276 C6MZ1J 46884121 IC50 = 1106 nM T80276 C96FTP 46884122 IC50 = 1478 nM T80276 C5RM6X 46884123 IC50 = 77 nM T80276 CKT35D 46884156 IC50 = 219 nM T80276 CFP9B5 46884157 IC50 = 36 nM T80276 CI3U2Q 46884158 IC50 = 49 nM T80276 CTVN70 46884203 IC50 = 57 nM T80276 C4FC9H 46884204 IC50 = 52 nM T80276 CEJ9C3 46884242 IC50 = 70 nM T80276 C8S5TR 46884243 IC50 = 100 nM T80276 CU93BN 46884282 IC50 = 25 nM T80276 C2H5CE 46884283 IC50 = 455 nM T80276 CWFH78 46884284 IC50 = 369 nM T80276 CZ5M8O 46884285 IC50 = 5895 nM T80276 CV3C0K 46884353 IC50 = 29 nM T80276 CZV8T9 46884354 IC50 = 155 nM T80276 CO9W8A 46884355 IC50 = 119 nM T80276 CLA01F 46884356 IC50 = 53 nM T80276 CO1D2H 46884404 IC50 = 104 nM T80276 CB6YM8 46884405 IC50 = 19 nM T80276 CL8PR5 46884406 IC50 = 173 nM T80276 CY9M0N 46884525 IC50 = 253 nM T80276 CH0QN3 46884526 IC50 = 1028 nM T80276 CAU6E8 46884527 IC50 = 2506 nM T80276 CA2U0D 46884528 IC50 = 4766 nM T80276 C5JBC1 46884529 IC50 = 592 nM T80276 CH2RD9 46884530 IC50 = 665 nM T80276 CWHK39 46884531 IC50 = 51 nM T80276 CSQ5I3 46884532 IC50 = 777 nM T80276 CS0Q3T 46884533 IC50 = 294 nM T80276 CO5H2J 46884534 IC50 = 574 nM T80276 C31KXQ 46884535 IC50 = 660 nM T80276 C86PXB 46884536 IC50 = 382 nM T80276 C6TI7E 46884537 IC50 = 79 nM T80276 CRW39C 46884538 IC50 = 77 nM T80276 C02IJK 46884539 IC50 = 54 nM T80276 C4SX6O 46884540 IC50 = 876 nM T80276 CE5S7W 46884541 IC50 = 286 nM T80276 CAS1R6 46884542 IC50 = 1006 nM T80276 C87UVQ 46884543 IC50 = 970 nM T80276 C2RJ4E 46884544 IC50 = 443 nM T80276 CE8YC5 46884545 IC50 = 102 nM T80276 CM3C9U 46884546 IC50 = 43 nM T80276 CGY1E3 46884547 IC50 = 610 nM T80276 CNW6L5 46884548 IC50 = 1896 nM T80276 CE12VC 46884549 IC50 = 644 nM T80276 CBR89Q 46884582 IC50 = 593 nM T80276 CK10UQ 46884583 IC50 = 173 nM T80276 CIJ4M5 46884584 IC50 = 846 nM T80276 CBD29C 46884585 IC50 = 330 nM T80276 CPE4I6 46884586 IC50 = 287 nM T80276 C09HUK 46884587 IC50 = 413 nM T80276 C8X3AD 46884588 IC50 = 314 nM T80276 CAHK18 46884589 IC50 = 76 nM T80276 CJZ75T 46884590 IC50 = 55 nM T80276 C1FXZ6 46884591 IC50 = 220 nM T80276 C0AD4G 46884592 IC50 = 414 nM T80276 CHF2L9 46884593 IC50 = 269 nM T80276 C1G6JK 46884594 IC50 = 402 nM T80276 CUPR76 46885272 IC50 = 52 nM T80276 CHP18Q 46885273 IC50 = 60 nM T80276 CY89OZ 46885274 IC50 = 947 nM T80276 CZ1XR9 46885275 IC50 = 1127 nM T80276 C9N5RS 46885276 IC50 = 499 nM T80276 CZYO07 46885277 IC50 = 226 nM T80276 C1Y7QN 46885278 IC50 = 955 nM T80276 CNLX49 46885279 IC50 = 483 nM T80276 CSA92E 46885280 IC50 = 389 nM T80276 CL4ZI9 46885281 IC50 = 961 nM T80276 CN3RH4 46885425 IC50 = 6754 nM T80276 CLA40T 46885426 IC50 = 492 nM T80276 COL95X 46885494 IC50 = 1889 nM T80276 CVWU94 46885495 IC50 = 3197 nM T80276 CC8T1E 46885496 IC50 = 179 nM T80276 CM8JX9 46885534 IC50 = 3650 nM T80276 CCS20H 46885565 IC50 = 1 nM T80276 CG47YP 46885566 IC50 = 106 nM T80276 C4R3XP 46885599 IC50 = 7 nM T80276 C3SMV1 46885600 IC50 = 2665 nM T80276 CV5MK6 46885601 IC50 = 36 nM T80276 C2M1DN 46885624 IC50 = 20 nM T80276 C42WVO 46885648 IC50 = 4 nM T80276 C0ZV8M 46886360 IC50 = 1 nM T80276 C1JS5T 46886361 IC50 = 5 nM T80276 CGRO36 46886375 IC50 < 1 nM T80276 CZR3V2 46886410 IC50 = 2 nM T80276 C4PRU3 46891423 IC50 = 0.4 nM T80276 CXPZ24 46891467 IC50 = 0.5 nM T80276 C9G4IW 46891468 IC50 = 0.4 nM T80276 C4IW0N 46891469 IC50 = 1 nM T80276 CF17MQ 46891470 IC50 = 0.2 nM T80276 CRHK80 46891471 IC50 = 0.2 nM T80276 C9SUH8 46891472 IC50 = 0.3 nM T80276 CGME41 46891473 IC50 = 0.5 nM T80276 C3HMQ2 46891474 IC50 = 0.2 nM T80276 CARY94 46891475 IC50 = 0.9 nM T80276 CB6Z8P 46892208 IC50 = 7700 nM T80276 CZX46Y 46892342 IC50 = 630 nM T80276 C5FN6I 46892845 IC50 = 798 nM T80276 CQ32BN 46892970 IC50 = 4 nM T80276 COJA32 46892971 Ki = 16 nM T80276 C5QFB3 46893088 IC50 = 200 nM T80276 C1Q8HJ 46893484 IC50 = 370 nM T80276 CO5ZE0 46893618 IC50 = 42 nM T80276 CS30AI 46893754 IC50 = 6200 nM T80276 CJK9Z8 46917909 IC50 = 36 nM T80276 CPO1N7 46927938 Ki = 1.77 nM T80276 CJ0VB4 46932297 IC50 = 14 nM T80276 CXZI94 46940004 IC50 = 89 nM T80276 CFO9X3 46946049 IC50 = 10 nM T80276 CL84AF 46946248 IC50 = 35 nM T80276 CF14PE 46947264 IC50 = 8 nM T80276 CV90JU 49764911 IC50 = 12589.25 nM T80276 COE37N 49778924 IC50 = 2500 nM T80276 CMRT49 49780177 IC50 > 300 nM T80276 C2Y9OC 49780178 IC50 > 300 nM T80276 C7ZK3D 49783923 IC50 = 501.19 nM T80276 CHX76J 49784892 Ki = 110 nM T80276 CA1H8S 49784893 Ki = 92 nM T80276 CP2QD0 49784894 Ki = 9 nM T80276 CTZG05 49784988 Ki = 200 nM T80276 CE9AC5 49785078 Ki = 190 nM T80276 CG2IO7 49785079 Ki = 39 nM T80276 C8EYN4 49785083 Ki = 100 nM T80276 CZI34V 49785167 Ki = 930 nM T80276 CJK65T 49785253 Ki = 28 nM T80276 CVU6P1 49785344 Ki = 2 nM T80276 CXK8F5 49785436 Ki = 5 nM T80276 CWL5C6 49785518 Ki = 8 nM T80276 C3NV0J 49785827 Ki = 12 nM T80276 C0OZM2 49785828 Ki = 61 nM T80276 C1AR4G 49785829 Ki = 1700 nM T80276 CA53NO 49788443 IC50 = 0.4 nM T80276 C2TRM0 49817355 IC50 = 75 nM T80276 C9ZW3R 49835055 IC50 = 590 nM T80276 CI6B7G 49835106 Ki = 29 nM T80276 CN2E0P 49835107 IC50 = 763 nM T80276 CV50DY 49835108 Ki = 14 nM T80276 CTM6U1 49835172 Ki = 6.3 nM T80276 CL6V8Y 49835227 IC50 = 256 nM T80276 C90XTJ 49835286 IC50 = 54 nM T80276 C5UR4A 49843944 IC50 = 130 nM T80276 CA4NH7 49850583 IC50 = 9000 nM T80276 CT4Y6E 49852123 IC50 > 50000 nM T80276 CS40YB 49853846 IC50 = 260 nM T80276 C0JV4U 49853889 IC50 = 6 nM T80276 C2EJ6Q 49853890 IC50 = 1044 nM T80276 C7PER0 49853953 IC50 = 25 nM T80276 CU9A8O 49854022 IC50 = 8510 nM T80276 C51QVH 49854023 IC50 = 4320 nM T80276 CM4HQ2 49854024 IC50 = 7610 nM T80276 C1LBX3 49854049 IC50 = 4 nM T80276 CVC2H6 49854052 IC50 = 6 nM T80276 CC2X9N 49854121 IC50 > 10000 nM T80276 CAJ58E 49854156 IC50 = 6 nM T80276 CAU39Y 49854158 IC50 = 4 nM T80276 CPK6X3 49854360 IC50 = 19 nM T80276 CBVT70 49854361 IC50 = 28 nM T80276 CQ1TZ6 49854365 IC50 = 70 nM T80276 CJ5I9X 49854461 IC50 = 10 nM T80276 CDXQ69 49854462 IC50 = 9 nM T80276 C0ORZ9 49854466 IC50 = 10 nM T80276 CV2I9K 49854502 IC50 = 743 nM T80276 CY14XF 49854572 IC50 = 5 nM T80276 CEC10T 49854573 IC50 = 4 nM T80276 C39KQW 49854679 IC50 = 5 nM T80276 C8VDR2 49854680 IC50 = 5 nM T80276 CN2V8R 49854681 IC50 = 10 nM T80276 CSN96A 49855001 IC50 = 19 nM T80276 CALY90 49855192 IC50 = 43 nM T80276 CJPE20 49855193 IC50 = 14 nM T80276 C1OM3I 49855237 IC50 = 3410 nM T80276 C26IQK 49857091 IC50 = 700 nM T80276 CR0PN9 49857092 IC50 = 10200 nM T80276 CCJN26 49857093 IC50 = 7200 nM T80276 C3YG5L 49857275 IC50 > 10000 nM T80276 CHO65B 49857279 IC50 = 5120 nM T80276 C9HMY1 49857280 IC50 = 66 nM T80276 CGW9L1 49857476 IC50 = 1000 nM T80276 CRD84P 49857479 IC50 = 700 nM T80276 COF78C 49857678 IC50 > 10000 nM T80276 C4H7XG 49857865 IC50 = 2200 nM T80276 CY8MP7 49867926 IC50 = 39 nM T80276 CR0IA5 49871864 IC50 > 20000 nM T80276 C13WJZ 49872243 IC50 = 1150 nM T80276 C5OY7B 49872246 IC50 = 703 nM T80276 C2KD5E 49872344 IC50 = 5080 nM T80276 CV5BF3 49872645 IC50 = 12600 nM T80276 CN97FO 49872646 IC50 = 949 nM T80276 CL64NB 49872737 IC50 = 6230 nM T80276 CRNG04 49872831 IC50 = 420 nM T80276 CQC8B4 49872835 IC50 = 1080 nM T80276 CPS3O1 49872924 IC50 = 1200 nM T80276 CUBX74 49872925 IC50 = 900 nM T80276 CAW69U 49872927 IC50 = 920 nM T80276 CV1L4P 49873242 IC50 = 5750 nM T80276 C5BA2V 49873243 IC50 = 10900 nM T80276 CSN45W 49873329 IC50 = 444 nM T80276 CPI56O 50908575 IC50 = 340 nM T80276 CP1D2X 50908576 IC50 = 400 nM T80276 C9CW7X 50908894 IC50 = 17 nM T80276 CJ8VL4 50925575 IC50 = 12 nM T80276 CD3H8X 50925576 IC50 = 12 nM T80276 CZK43Y 50925577 IC50 = 31 nM T80276 CJ4L8Y 50938829 Ki > 125000 nM T80276 CJG65L 50939078 Ki = 3250 nM T80276 CI8QM1 50939080 Ki = 510 nM T80276 CT0IP3 50939081 Ki = 3540 nM T80276 C54EUL 50939212 Ki > 12500 nM T80276 CS7Z6U 50939338 Ki = 1720 nM T80276 C2I9PS 50939992 IC50 = 41000 nM T80276 C9TUE4 50940108 IC50 = 2320 nM T80276 C25YNT 50940492 Ki = 1 nM T80276 C2Q0GE 50990922 IC50 = 320 nM T80276 CKY3V1 50990924 Ki = 1.2 nM T80276 C5ZF9W 51003380 IC50 = 10200 nM T80276 CGQ49I 51003483 Ki = 7 nM T80276 C0HWJ7 51003484 Ki = 15 nM T80276 CHP3Z4 51003485 Ki = 0.5 nM T80276 CXD71B 51003497 IC50 = 70 nM T80276 CY36EH 51003592 IC50 = 794.33 nM T80276 CPA8N1 51039139 Ki > 10000 nM T80276 CLB85F 51346892 IC50 = 140 nM T80276 C65ILG 51346893 IC50 = 62 nM T80276 CQ6DM8 51347750 Ki = 0.14 nM T80276 C3P7EZ 51348054 Ki = 0.11 nM T80276 CIY2Q6 51350683 EC50 > 1250 nM T80276 C90AZG 51350684 EC50 = 1000 nM T80276 CN7R6E 51350805 EC50 = 250 nM T80276 CD56KO 51350806 EC50 = 500 nM T80276 CM36TE 51350807 EC50 = 500 nM T80276 CV2JN5 51350808 EC50 = 750 nM T80276 CUL3F1 51350809 EC50 = 1000 nM T80276 CKD86C 51350810 EC50 > 1250 nM T80276 C8A7LY 51350918 EC50 = 1000 nM T80276 C05XQL 51350919 EC50 = 1000 nM T80276 CP93ZQ 51350921 EC50 > 1250 nM T80276 CBV7T1 51350922 EC50 = 250 nM T80276 C5R0SE 51350923 EC50 = 500 nM T80276 C7EVF8 51351030 EC50 = 1000 nM T80276 CD0RS6 51351031 EC50 = 750 nM T80276 CSD65R 51351032 EC50 = 750 nM T80276 C38WSA 51351033 EC50 = 250 nM T80276 C4E6BY 51351034 EC50 = 750 nM T80276 C6B1JI 51351035 EC50 = 1000 nM T80276 C2VPD0 51351157 EC50 > 1250 nM T80276 C8FOH4 51351158 EC50 = 1250 nM T80276 CVK96A 51351159 EC50 = 1250 nM T80276 CLZ8N6 51352027 IC50 = 794.33 nM T80276 C73ANH 51353707 Ki = 117 nM T80276 CI4A6R 51353708 Ki = 76 nM T80276 CJ4ZL6 51353709 Ki = 62 nM T80276 CDLF71 51353710 Ki = 41 nM T80276 C04EVK 51353711 Ki = 65 nM T80276 CD6AL8 51353712 Ki = 84 nM T80276 CPQ1G6 51354021 Ki = 826 nM T80276 CVK95R 51354022 Ki = 82 nM T80276 CHKA96 51354023 Ki = 38 nM T80276 CRL1B8 51354025 Ki = 3130 nM T80276 C6VD0B 51354313 Ki = 13 nM T80276 CJC90Y 51354315 Ki = 1.6 nM T80276 COH9L7 51354317 Ki = 9 nM T80276 CV6I5D 51354595 Ki = 48 nM T80276 C1V6RN 51354597 Ki = 1.4 nM T80276 CZ32XV 51354599 Ki = 1.2 nM T80276 C8WEN4 51354600 Ki < 1 nM T80276 C76KOV 51354878 Ki < 1 nM T80276 CA3O2L 51354879 Ki < 1 nM T80276 C0O2PW 51354880 Ki < 1 nM T80276 C3JV4L 51354881 Ki < 1 nM T80276 C6NL1Z 51354882 Ki < 1 nM T80276 CPWD73 51354883 Ki < 1 nM T80276 C6E9WP 51355057 Ki > 10000 nM T80276 C4QE1V 51355058 IC50 = 5800 nM T80276 CB10AP 51355171 Ki < 1 nM T80276 CKE42Q 51355172 Ki < 1 nM T80276 CZF89J 51355173 Ki < 1 nM T80276 CQF0J9 51355174 Ki = 1.1 nM T80276 CO7M9F 51355343 IC50 > 10000 nM T80276 CJ0KM6 51355344 IC50 = 6400 nM T80276 CT0V8F 51355345 Ki > 10000 nM T80276 C0R8XN 51355348 Ki = 5800 nM T80276 C7KT4Z 51355620 Ki = 3400 nM T80276 CI71WE 51355621 Ki = 5135 nM T80276 CLH35Z 51355622 Ki = 7000 nM T80276 C2ODW5 51357942 Ki = 6100 nM T80276 CSR12N 51357943 Ki = 1010 nM T80276 CT8LF4 51357944 Ki = 31 nM T80276 C8IOD1 51357945 Ki = 47 nM T80276 C1KB9V 51357946 Ki = 18 nM T80276 C7HOD9 51357947 Ki = 58 nM T80276 CI7MJ6 51357948 Ki = 24 nM T80276 CRJ5W8 51358113 EC50 = 200 nM T80276 CT91WR 52040626 IC50 > 1000 nM T80276 CD84MT 52913592 IC50 = 130 nM T80276 C2TLG6 52913931 IC50 = 170 nM T80276 C7P2IG 52936736 IC50 = 5200 nM T80276 CM0AO4 52936737 IC50 = 360 nM T80276 C9HS0D 52936847 IC50 = 2 nM T80276 CNZ87U 52936848 IC50 = 11 nM T80276 CVQ76Y 52936850 IC50 = 2 nM T80276 CVDI14 52936957 IC50 = 213 nM T80276 CE0K9Q 52936958 IC50 = 0.8 nM T80276 CTZ47U 52936959 IC50 = 36 nM T80276 CR16NY 52936960 IC50 = 720 nM T80276 CVD2W7 52936961 IC50 = 12 nM T80276 CYOJ94 52936962 IC50 = 7 nM T80276 CWL9C1 52937061 IC50 = 4 nM T80276 CUN68K 52937062 IC50 = 47 nM T80276 CJO4M9 52937063 IC50 = 480 nM T80276 CK7Z9W 52937064 IC50 = 10 nM T80276 C36UMZ 52937065 IC50 = 2 nM T80276 CS1TE9 52937066 IC50 = 0.6 nM T80276 CRCD47 52937166 IC50 = 81 nM T80276 CU1P2L 52940797 IC50 = 1370 nM T80276 CD62QJ 52940982 IC50 = 13.5 nM T80276 C9N7GZ 52941270 IC50 = 11 nM T80276 CI6VH8 52941280 IC50 = 15000 nM T80276 C43SVQ 52941322 IC50 = 21 nM T80276 C1HO7N 52941331 IC50 = 1100 nM T80276 CK59HM 52941479 IC50 = 17 nM T80276 C8U7XA 52941692 IC50 = 16 nM T80276 C2KI6V 52942202 IC50 = 10000 nM T80276 CDHJ08 52942235 IC50 = 2600 nM T80276 C54LPV 52942609 IC50 = 1300 nM T80276 C68RNX 52942729 IC50 = 5600 nM T80276 CFRN73 52942850 IC50 = 69 nM T80276 C4D1KT 52942879 IC50 = 40 nM T80276 C4VCY0 52943258 IC50 = 29000 nM T80276 C1XEV2 52943394 IC50 = 3680 nM T80276 C73WTL 52943744 IC50 = 21 nM T80276 C6Q1AH 52943745 IC50 = 14 nM T80276 C4WB7S 52943856 IC50 = 730 nM T80276 CHIG53 52943884 IC50 = 570 nM T80276 C98KZO 52943947 IC50 = 16000 nM T80276 CHI0P6 52944356 IC50 = 100000 nM T80276 C69WST 52944867 IC50 = 9400 nM T80276 CCH9V6 52944935 IC50 = 1.7 nM T80276 C7F3KG 52945072 IC50 = 430 nM T80276 CWD27C 52945142 IC50 = 84 nM T80276 CAX50E 52945171 IC50 = 15000 nM T80276 CWPC54 52945348 IC50 = 450 nM T80276 CXL53B 52945589 IC50 = 39 nM T80276 C4NLX7 52945630 IC50 = 433 nM T80276 CXD6T8 52945845 IC50 = 3400 nM T80276 C3N6PO 52946107 IC50 = 13000 nM T80276 CH2IQ4 52946207 IC50 = 1.1 nM T80276 C54FIO 52946229 IC50 = 620 nM T80276 CX4P8A 52946248 IC50 = 720 nM T80276 CN8F0V 52946289 IC50 = 3.5 nM T80276 CMQY93 52946368 IC50 = 28 nM T80276 C8R0AS 52946467 IC50 = 11000 nM T80276 C54LRW 52947235 IC50 > 300 nM T80276 C0W2MY 52947387 IC50 = 14000 nM T80276 CE7BL1 52947388 IC50 = 16000 nM T80276 C07RTQ 52947480 IC50 = 50 nM T80276 C4DV1W 52947519 IC50 = 950 nM T80276 CET7P0 52947556 IC50 = 130 nM T80276 CXO3V9 52947717 IC50 = 190 nM T80276 C5X9VO 52948007 IC50 = 86 nM T80276 C7ET6Z 52948010 IC50 = 1300 nM T80276 C5CXZ3 52948541 IC50 = 9500 nM T80276 CIS71L 52948791 IC50 = 134 nM T80276 C5PFI4 52948798 IC50 = 3 nM T80276 C20FHZ 52948848 IC50 = 3640 nM T80276 CN84EL 52948997 IC50 = 11000 nM T80276 CW9Z1T 52949347 IC50 = 18 nM T80276 CS1TG3 52949440 IC50 = 56 nM T80276 CV5B2C 52949497 IC50 = 100000 nM T80276 CB0KM5 52949869 IC50 = 7 nM T80276 CAJQ03 52950001 IC50 = 23 nM T80276 CBZP60 52950005 IC50 = 72 nM T80276 CE6L8W 52950012 IC50 = 460 nM T80276 C7MC1H 52950013 IC50 = 1600 nM T80276 CPW0H2 52950026 IC50 = 7800 nM T80276 CN90FO 52950046 IC50 = 386 nM T80276 C5HQ2E 52950102 IC50 = 14 nM T80276 CH1Q5D 53234281 IC50 = 3.1 nM T80276 C45JKN 53234283 IC50 = 99 nM T80276 CVK28S 53235062 IC50 < 0.5 nM T80276 C9PF3V 53235144 IC50 = 1.3 nM T80276 COW61E 53235216 IC50 = 2 nM T80276 CWE56X 53235217 IC50 = 1.4 nM T80276 CE80SC 53235449 IC50 = 3.3 nM T80276 CDXM59 53235451 IC50 = 11 nM T80276 CT8IN1 53242225 IC50 = 2200 nM T80276 C4J9WZ 53307606 Ki = 2 nM T80276 C8N5BU 53316474 IC50 = 290 nM T80276 CT54XZ 53316658 Ki = 6 nM T80276 CRD3A9 53316967 IC50 = 260 nM T80276 CG6O0M 53317018 Ki = 188 nM T80276 C84YNK 53317325 IC50 = 29300 nM T80276 CBOR03 53317408 IC50 > 10000 nM T80276 CSV3I8 53317409 IC50 > 10000 nM T80276 C2CNP7 53317512 IC50 = 774 nM T80276 C42HGW 53317513 EC50 = 110 nM T80276 CW8PM0 53317812 IC50 = 3000 nM T80276 CS8DJ3 53318252 IC50 = 140 nM T80276 C8FPQ4 53318293 Ki = 100 nM T80276 C2KP0W 53318294 Ki = 100 nM T80276 CK9SE2 53318295 Ki = 5 nM T80276 C58NQJ 53318614 IC50 > 83300 nM T80276 C10YUH 53318615 IC50 = 13000 nM T80276 CDU61K 53318702 IC50 > 10000 nM T80276 CJ81GS 53318703 IC50 > 10000 nM T80276 CT35VY 53318704 IC50 = 770 nM T80276 CQ7FO6 53318739 IC50 = 1000 nM T80276 C32YWC 53318782 IC50 = 13 nM T80276 CCP80W 53319118 IC50 = 150 nM T80276 CFJD70 53319932 IC50 = 59000 nM T80276 C3EJB1 53319933 IC50 = 10800 nM T80276 C2V7AX 53320017 IC50 = 180 nM T80276 CKGJ60 53320018 IC50 = 110 nM T80276 C4LIJ2 53320019 IC50 > 10000 nM T80276 C4Q1AO 53320102 EC50 = 370 nM T80276 CFSA29 53320103 EC50 = 390 nM T80276 C65GKX 53320104 IC50 = 44 nM T80276 C3Z4FD 53320358 IC50 = 1600 nM T80276 CA2QV6 53320444 IC50 = 430 nM T80276 C7C4LR 53320445 IC50 = 1100 nM T80276 C6T3BN 53320905 IC50 = 200 nM T80276 CMT3N2 53320906 IC50 = 1000 nM T80276 C7WQ3Z 53320907 IC50 = 860 nM T80276 C1EQ6B 53321327 IC50 = 660 nM T80276 CV7EI8 53321328 IC50 > 10000 nM T80276 CFW30O 53321329 IC50 > 10000 nM T80276 C3AN0K 53321330 IC50 = 9100 nM T80276 C46YVK 53321409 IC50 = 55 nM T80276 CQRU94 53321410 IC50 = 66 nM T80276 C27AWP 53321743 IC50 = 4400 nM T80276 CY8DH9 53322283 Ki = 54 nM T80276 CJRM64 53322563 IC50 = 22700 nM T80276 CFSU71 53322641 IC50 = 1300 nM T80276 CJ7GQ2 53322730 IC50 = 253 nM T80276 CO0K3S 53322731 IC50 < 2 nM T80276 CN92LK 53322732 IC50 < 2 nM T80276 CIN6Q4 53322733 IC50 = 6 nM T80276 C0R6BV 53322917 IC50 = 6200 nM T80276 CLX39O 53323075 IC50 = 150 nM T80276 CCP53L 53323076 IC50 = 1500 nM T80276 CP15UQ 53323077 IC50 = 290 nM T80276 CIJ0K1 53323078 IC50 = 270 nM T80276 CMDJ03 53323585 IC50 > 10000 nM T80276 C7RW4X 53323586 IC50 > 10000 nM T80276 CCSP27 53323641 Ki = 0.5 nM T80276 CW9F1T 53323642 Ki = 12 nM T80276 CQX59J 53323643 Ki = 631 nM T80276 C03WPK 53323982 IC50 = 250 nM T80276 CJG3R2 53323983 IC50 = 230 nM T80276 CDI05T 53323984 IC50 = 1100 nM T80276 CTD8A0 53324021 Ki = 4550 nM T80276 CYCB54 53324065 EC50 = 650 nM T80276 CVDR80 53324066 EC50 = 450 nM T80276 C3JYD5 53324329 IC50 < 2 nM T80276 C7TR8E 53324425 IC50 = 350 nM T80276 C69PLZ 53324426 IC50 = 470 nM T80276 CENI79 53324886 IC50 > 10000 nM T80276 C85XMQ 53324887 IC50 = 690 nM T80276 CJ7A6D 53324888 IC50 = 880 nM T80276 CZ41DR 53324923 Ki = 4550 nM T80276 CPYO04 53325279 IC50 > 10000 nM T80276 CWO65H 53325280 IC50 > 10000 nM T80276 CVDH70 53325281 IC50 = 8900 nM T80276 C51VYQ 53325282 IC50 = 440 nM T80276 CDX13C 53325373 IC50 > 10000 nM T80276 CJZ29M 53325374 IC50 = 250 nM T80276 C1TE8J 53325515 IC50 = 900 nM T80276 C4CU5V 53325726 IC50 = 400 nM T80276 CPW9G1 53326165 IC50 > 10000 nM T80276 C6LAI9 53326166 IC50 = 260 nM T80276 CZQ80X 53326214 Ki = 0.5 nM T80276 CA3SF4 53326215 Ki = 100 nM T80276 C25LHM 53326216 Ki = 0.3 nM T80276 C87JDW 53326551 IC50 = 860 nM T80276 CFAX51 53326552 IC50 > 10000 nM T80276 CMFL35 53326553 IC50 = 820 nM T80276 CD70CU 53326636 IC50 = 247 nM T80276 C8D5SQ 53326637 EC50 = 130 nM T80276 CGC6N0 53326793 IC50 = 500 nM T80276 CUYM86 53326857 IC50 = 300 nM T80276 CT5V9I 53326947 IC50 = 1350 nM T80276 CRYW35 53350231 Ki = 1 nM T80276 C23HAU 53361718 Ki = 0.7 nM T80276 CM60WQ 53361719 Ki = 0.8 nM T80276 CBPR36 53363353 Ki = 12.9 nM T80276 C21UXP 53363435 Ki = 2.6 nM T80276 C50DRH 53363439 Ki = 69 nM T80276 CQT13C 53363523 Ki = 0.7 nM T80276 C9WMI6 53363529 Ki = 1.7 nM T80276 CV9L6P 53363611 Ki = 1 nM T80276 CL69DK 53377727 IC50 = 7 nM T80276 C6Q8RC 53378051 IC50 = 1258.93 nM T80276 CG3C1J 53379513 IC50 = 0.2 nM T80276 CP4W1Q 53380858 IC50 = 6309.57 nM T80276 C5SMC3 53387410 Ki = 6.1 nM T80276 C5Q0HA 53387411 Ki = 23 nM T80276 C90KZU 53387571 Ki = 119 nM T80276 CMO9K1 53387572 Ki = 68 nM T80276 CI40BG 53387573 Ki = 7.2 nM T80276 C2IJR7 53387574 Ki = 26 nM T80276 CWB79U 53387575 Ki = 51 nM T80276 CB4H9G 53387738 Ki = 47 nM T80276 C5ZY9R 53387740 Ki = 76 nM T80276 CVG90B 53389651 IC50 > 10000 nM T80276 CSV9X2 54579940 IC50 = 6 nM T80276 CN51TL 54579941 IC50 = 6200 nM T80276 C7VZU2 54579942 IC50 = 840 nM T80276 C4R9JB 54579943 IC50 = 460 nM T80276 CG26HQ 54579944 IC50 = 4000 nM T80276 CQE1Z7 54580062 IC50 = 340 nM T80276 C5O9WP 54580063 IC50 = 520 nM T80276 CC5R3O 54580924 IC50 = 230 nM T80276 C3OIY4 54580925 IC50 = 490 nM T80276 CUP7N6 54581023 IC50 = 720 nM T80276 CAB63J 54581048 IC50 = 2000 nM T80276 C60TYL 54581049 IC50 = 260 nM T80276 CF2UH5 54581983 IC50 = 23 nM T80276 CB3OM9 54582056 IC50 = 3600 nM T80276 C5B4MV 54582091 IC50 = 1000 nM T80276 C23EVN 54582916 IC50 = 520 nM T80276 CT2SV7 54583916 IC50 = 290 nM T80276 CY87EC 54583917 IC50 = 1600 nM T80276 C2GE8J 54584039 IC50 = 3600 nM T80276 CT3CN8 54584240 EC50 > 1250 nM T80276 C8CPI4 54584859 IC50 = 10400 nM T80276 C9TZ2V 54584860 IC50 = 1900 nM T80276 CVY42B 54584949 IC50 = 190 nM T80276 C1M9JE 54584986 IC50 = 1700 nM T80276 CME81Q 54585830 IC50 = 960 nM T80276 C81YUR 54585940 IC50 = 130 nM T80276 CW95OA 54586162 EC50 > 1250 nM T80276 C1G0IY 54586917 IC50 = 3500 nM T80276 CQE3L1 54669876 Ki = 3 nM T80276 CFI7E6 54754350 IC50 = 25 nM T80276 C0Y9ZG 54761473 IC50 > 30000 nM T80276 CU8YW6 56325569 IC50 = 55000 nM T80276 CE4TS9 56589559 IC50 = 4.8 nM T80276 CR24WQ 56595421 IC50 = 3 nM T80276 CJ41GT 56595686 IC50 = 49 nM T80276 C2PN4S 56599298 IC50 = 1940 nM T80276 CT64SR 56599306 IC50 = 39 nM T80276 CFUT05 56648675 IC50 = 0.7 nM T80276 C1GAB6 56648677 IC50 = 2.1 nM T80276 CWDF40 56648757 IC50 = 1 nM T80276 CE35CB 56648758 Ki = 2.8 nM T80276 CJO39U 56648759 IC50 = 1.7 nM T80276 CNKC90 56654649 IC50 = 590 nM T80276 CCR56D 56659711 IC50 = 5200 nM T80276 C83QGP 56660108 IC50 = 0.6 nM T80276 CYM1D0 56660109 IC50 = 1.4 nM T80276 CY5F7J 56663363 IC50 > 1000 nM T80276 CHA35L 56663573 IC50 = 1.4 nM T80276 CF7PY5 56667023 IC50 = 0.4 nM T80276 CL5KG7 56670030 IC50 = 1000 nM T80276 CCH69F 56670031 IC50 = 17000 nM T80276 CC1DJ8 56670464 IC50 = 2 nM T80276 C2MDB8 56673545 IC50 > 10000 nM T80276 CE2Q5Y 56673546 Ki = 1 nM T80276 CZH95G 56673952 IC50 = 1.4 nM T80276 CY95CZ 56676870 IC50 = 673 nM T80276 C2DZR0 56677061 IC50 = 470 nM T80276 CHR8K0 56677282 IC50 = 0.6 nM T80276 C79AMB 56677283 IC50 = 1.2 nM T80276 CQME43 56680186 Ki = 16 nM T80276 CL68MS 56680202 Ki = 65 nM T80276 C2ZAF3 56680380 IC50 = 70 nM T80276 CUN09R 56680409 IC50 > 1000 nM T80276 C5ZN6X 56682067 Ki = 5.6 nM T80276 CXI9Y4 56683527 IC50 > 10000 nM T80276 CY82AC 56683542 Ki = 473 nM T80276 C4PXD1 56683543 Ki = 2.5 nM T80276 CQ6Z0N 56683747 IC50 > 1000 nM T80276 CG17TZ 56683916 IC50 = 0.8 nM T80276 C7B2OH 56683917 IC50 = 1 nM T80276 C6LMP8 56683918 IC50 = 1.7 nM T80276 C94JIT 56832510 Ki = 0.27 nM T80276 CC9IP6 56833458 Ki = 1 nM T80276 CKD9T4 56833539 Ki = 47 nM T80276 CLG1W9 56833540 Ki = 9 nM T80276 C7GMY3 56833541 Ki = 5 nM T80276 CI0LP9 56833542 Ki = 2 nM T80276 CE2XW4 56833543 Ki = 0.4 nM T80276 C6PK0Z 56833544 Ki = 1 nM T80276 C07XMA 56833636 Ki = 1 nM T80276 C7RA0U 56833637 Ki = 3 nM T80276 CBHQ53 56833638 Ki = 4 nM T80276 CY7Q6N 56833639 Ki = 4 nM T80276 CPDO94 56833738 Ki = 1 nM T80276 C5C6QT 56833739 Ki = 1 nM T80276 CK36WM 56833740 Ki = 48 nM T80276 CNP72B 56834968 IC50 = 33.6 nM T80276 CH92MC 56834969 IC50 = 49.7 nM T80276 CLX13D 56834970 IC50 = 60.7 nM T80276 CNBS48 56834971 IC50 = 47.8 nM T80276 C0IJP8 56927258 IC50 = 1584.89 nM T80276 C9MJG4 56929824 EC50 < 40 nM T80276 CYFB96 56932203 IC50 > 6309.57 nM T80276 CJ9R2C 56932209 IC50 = 3981.07 nM T80276 C8C2FG 56932238 IC50 > 19952.62 nM T80276 CX6Q2K 56932240 IC50 = 3162.28 nM T80276 C0M3EQ 56950791 IC50 = 1100 nM T80276 CO6K5Q 56955953 IC50 = 960 nM T80276 CAK91L 56955954 IC50 = 435 nM T80276 C8B6JG 56955955 IC50 = 505 nM T80276 C74YNV 56966983 IC50 = 13.1 nM T80276 CW8B4D 57330208 IC50 = 7900 nM T80276 C6JMN9 57345685 IC50 = 800 nM T80276 CZ7RE0 57345686 IC50 = 2000 nM T80276 CA53SC 57351276 Ki = 122 nM T80276 C3CL8H 57384862 Ki = 2 nM T80276 C1X3UP 57390135 IC50 > 1000 nM T80276 CQ6N8D 57390136 IC50 = 30 nM T80276 C6XDC8 57390137 IC50 = 610 nM T80276 C0S6IG 57390138 IC50 = 4.5 nM T80276 C2RI4V 57390139 IC50 > 1000 nM T80276 CZ3FU2 57390175 IC50 > 1000 nM T80276 CR2X7O 57390176 IC50 = 1600 nM T80276 C3NZL6 57391047 IC50 = 424.7 nM T80276 C1GVK3 57391362 IC50 = 5000 nM T80276 CLHX38 57391363 IC50 = 1600 nM T80276 C0PR9J 57391364 IC50 > 1300 nM T80276 C6L9HO 57391365 IC50 = 1000 nM T80276 C2QX0T 57391366 IC50 = 630 nM T80276 CLQ9J1 57391367 IC50 = 790 nM T80276 C53HZJ 57391915 IC50 = 1100 nM T80276 CO18UJ 57391916 IC50 = 7 nM T80276 CRU8Q0 57391917 IC50 = 80 nM T80276 C13DRO 57391952 IC50 > 1000 nM T80276 CH8UV4 57391962 IC50 = 1.5 nM T80276 CQ1W0C 57393124 IC50 > 4000 nM T80276 CZ0RW2 57393125 IC50 > 3200 nM T80276 C3G9VK 57393643 IC50 > 1000 nM T80276 CJX56V 57393644 IC50 = 2.4 nM T80276 CAND02 57393679 IC50 > 1000 nM T80276 CA93ZE 57394864 IC50 > 2000 nM T80276 CF6C2T 57395364 IC50 > 1000 nM T80276 CKE35B 57395365 IC50 = 39 nM T80276 CWL2D6 57395366 IC50 > 1000 nM T80276 CB6L7N 57395397 IC50 > 1000 nM T80276 CJH9S2 57395408 IC50 = 100 nM T80276 C31MCE 57395409 IC50 = 1.8 nM T80276 CSP45C 57395410 IC50 = 2.2 nM T80276 CDG2F3 57396625 IC50 = 630 nM T80276 CD73TE 57396626 IC50 = 6300 nM T80276 CQRU75 57396627 IC50 = 3200 nM T80276 CI34XH 57396628 IC50 > 4000 nM T80276 C92FYK 57397192 IC50 = 27 nM T80276 CBC7N6 57397236 IC50 > 1000 nM T80276 CK01SI 57397253 IC50 = 0.5 nM T80276 C4N7MX 57397773 IC50 > 30000 nM T80276 C2VPR0 57397894 IC50 = 21900 nM T80276 C26LFR 57398107 IC50 = 421.3 nM T80276 CU9N1Z 57398248 IC50 = 4050 nM T80276 C3Q2ZP 57398390 IC50 > 4000 nM T80276 C56TEZ 57398391 IC50 = 4000 nM T80276 CP9Q4U 57398392 IC50 = 4000 nM T80276 C0O5KE 57398393 IC50 = 800 nM T80276 C5PI3B 57398894 IC50 = 390 nM T80276 COTK97 57398895 IC50 > 1000 nM T80276 CD5Z7P 57399042 IC50 = 28 nM T80276 C3G9HW 57399126 IC50 > 4000 nM T80276 CLP47I 57399764 IC50 = 510.5 nM T80276 CYE09F 57400062 IC50 > 4000 nM T80276 CN5PY7 57400063 IC50 > 4000 nM T80276 CT0Y7E 57400064 IC50 = 1000 nM T80276 C0PZM5 57400579 IC50 = 1200 nM T80276 C9BW8C 57400580 IC50 = 14 nM T80276 C4K2RZ 57400581 IC50 > 1000 nM T80276 C4MW8J 57400582 IC50 > 1000 nM T80276 CGC91E 57400641 IC50 = 0.8 nM T80276 C7UYA9 57401258 IC50 > 30000 nM T80276 C0LP7R 57401331 IC50 > 30000 nM T80276 CM63CS 57401865 IC50 = 500 nM T80276 CG6M4H 57401867 IC50 = 5000 nM T80276 CP8FY5 57401868 IC50 = 1600 nM T80276 CQ5P4X 57401869 IC50 = 1600 nM T80276 C2X8PO 57402386 IC50 = 45 nM T80276 CNMV98 57402387 IC50 = 2.4 nM T80276 C06IYP 57402428 IC50 = 13 nM T80276 CWV56Z 57402952 IC50 > 30000 nM T80276 C5TPX8 57403086 IC50 = 23500 nM T80276 C3Q1CB 57403282 IC50 = 544 nM T80276 CF68RN 57403576 IC50 = 3200 nM T80276 CL2R7T 57403577 IC50 > 4000 nM T80276 CC5N9R 57403578 IC50 > 13000 nM T80276 CZ8M5F 57403579 IC50 > 4000 nM T80276 C5NT7R 57403580 IC50 = 790 nM T80276 CHBV63 57403581 IC50 = 400 nM T80276 CAC72X 57403582 IC50 > 3900 nM T80276 CNR95F 57404840 IC50 = 6800 nM T80276 COAT54 57406937 IC50 = 567 nM T80276 CED47A 57410062 IC50 = 1119 nM T80276 C1BVX6 57411134 IC50 = 4075 nM T80276 C39JSW 57411135 IC50 = 8280 nM T80276 CL8F6Q 57411137 IC50 > 10000 nM T80276 CW97FT 57411139 IC50 = 7230 nM T80276 CU0R3A 57411250 IC50 > 10000 nM T80276 C6C5TU 57411252 IC50 > 10000 nM T80276 CD0W2I 57411254 IC50 = 2146 nM T80276 CW1DA3 57411255 IC50 > 10000 nM T80276 C6U4LO 57411256 IC50 = 6968 nM T80276 CP9G7L 57411366 IC50 > 10000 nM T80276 CC5DO3 57411369 IC50 = 2208 nM T80276 C56RBS 57411372 IC50 = 6333 nM T80276 CX9O3T 57411485 IC50 > 10000 nM T80276 CQBM65 57411486 IC50 > 10000 nM T80276 CK5QX7 57411488 IC50 > 10000 nM T80276 C90LNK 57411715 IC50 > 10000 nM T80276 CPXE40 57411716 IC50 > 10000 nM T80276 CE6RY5 57411836 IC50 > 10000 nM T80276 C5JOX3 57411837 IC50 > 10000 nM T80276 C0I5JM 57419280 IC50 > 5000 nM T80276 CNI79K 57427669 IC50 = 7943.28 nM T80276 C8Y7VZ 57427751 IC50 = 7943.28 nM T80276 CK6TN2 57427752 IC50 = 3235.94 nM T80276 CT6XL0 57466811 Ki = 1400 nM T80276 CRB5P2 57495287 IC50 = 792 nM T80276 C59YAC 57495353 IC50 = 244 nM T80276 CMT9L7 57495355 IC50 = 651 nM T80276 CWQ6F2 57523291 IC50 > 10000 nM T80276 CJE19S 57523686 IC50 > 10000 nM T80276 CR1P7W 57598055 IC50 > 10000 nM T80276 CV9J7D 57748162 IC50 = 19 nM T80276 CL57CP 57789333 IC50 = 80 nM T80276 C81BYH 57798309 IC50 = 1500 nM T80276 CG1E3X 57900125 IC50 = 7 nM T80276 C0F1AG 57900132 IC50 < 0.5 nM T80276 C05ZNP 57900198 IC50 < 0.5 nM T80276 CV1NI8 57900240 IC50 < 0.5 nM T80276 CIB30V 57900255 IC50 = 8 nM T80276 CE78IO 57900289 IC50 = 7 nM T80276 CZ21KP 57900314 IC50 = 4 nM T80276 CU84KP 57900315 IC50 = 1.2 nM T80276 CGX2N9 57900394 IC50 = 279 nM T80276 CUAE94 57900409 IC50 = 1 nM T80276 CV1ET6 57900418 IC50 = 481 nM T80276 CVP5T2 57900428 IC50 < 0.5 nM T80276 CERT48 57900437 IC50 = 7.3 nM T80276 CHOC46 57900447 IC50 = 15 nM T80276 CY5BX9 57900462 IC50 = 1.2 nM T80276 CWXH46 57900475 IC50 = 142 nM T80276 CJF3U1 57900505 IC50 < 0.5 nM T80276 CJ9ZW8 57900523 IC50 < 0.5 nM T80276 C1EP6I 58024825 IC50 > 100000 nM T80276 C46AUK 58137055 IC50 = 980 nM T80276 C7ONC3 58137106 IC50 = 3800 nM T80276 C6DH9J 58137111 IC50 > 90000 nM T80276 C7VSX2 58137137 IC50 = 2050 nM T80276 C84FUI 58137148 IC50 = 36700 nM T80276 C5IMD7 58137170 IC50 = 7600 nM T80276 CRPL37 58137176 IC50 = 1060 nM T80276 CV7YP2 58169819 IC50 = 79.43 nM T80276 CJ8TE4 58169820 IC50 = 1258.93 nM T80276 C8S7NQ 58203695 Ki = 0.18 nM T80276 CO20YT 58203712 IC50 = 1.3 nM T80276 CINT74 58203776 Ki = 0.13 nM T80276 C7X0OJ 58203779 IC50 = 2 nM T80276 C36IVB 58203785 Ki = 0.15 nM T80276 C61ZNP 58203789 Ki = 0.94 nM T80276 CF85YJ 58203795 Ki = 0.11 nM T80276 CEM32T 58203808 Ki = 0.9 nM T80276 C5KLV8 58203898 Ki = 0.06 nM T80276 CG65RS 58203922 Ki = 0.69 nM T80276 CW1M9X 58203976 IC50 = 4.9 nM T80276 COFN62 58203995 IC50 = 3.5 nM T80276 CN8D9F 58204007 Ki = 0.18 nM T80276 CPDQ83 58204017 Ki = 0.06 nM T80276 C16GRS 58204034 IC50 = 364 nM T80276 CM62NB 58204076 IC50 < 0.5 nM T80276 C07NXV 58204082 Ki = 0.61 nM T80276 C81XIQ 58204138 Ki = 0.04 nM T80276 C8Y4RB 58204237 Ki = 1.9 nM T80276 CGA01N 58204242 IC50 = 1.5 nM T80276 C4MK5I 58204259 Ki = 0.47 nM T80276 C42SJN 58204320 Ki = 21.1 nM T80276 CPU5G7 58204339 Ki = 0.29 nM T80276 CSV27U 58204369 Ki = 3.6 nM T80276 CCGA59 58204388 Ki = 0.5 nM T80276 CGN08U 58204405 Ki = 1.2 nM T80276 CF31TC 58204526 IC50 = 33 nM T80276 CG5WR2 58204531 Ki = 0.1 nM T80276 C9TE0A 58204549 Ki = 0.1 nM T80276 C82WIV 58204557 Ki = 3.1 nM T80276 CV76WN 58204592 Ki = 0.03 nM T80276 C4WZ6M 58204628 Ki = 0.17 nM T80276 CN5K6L 58204658 IC50 = 3.3 nM T80276 CEN68J 58204703 Ki = 0.34 nM T80276 CVC76I 58204711 Ki = 0.4 nM T80276 CDYB40 58204717 Ki = 0.31 nM T80276 C30CFN 58204750 Ki = 30 nM T80276 CSD7W0 58204759 Ki = 0.3 nM T80276 CLP19A 58204821 Ki = 1.3 nM T80276 CE94DM 58204847 Ki = 0.2 nM T80276 CIQN06 58204851 Ki = 2.8 nM T80276 C9TH7I 58204871 Ki = 3.6 nM T80276 C81STA 58204873 Ki = 0.3 nM T80276 C6ZO1X 58204890 Ki = 0.9 nM T80276 CW3Q0T 58204894 Ki = 3.2 nM T80276 CSC46N 58204974 Ki < 1 nM T80276 CB72QI 58204997 Ki = 0.2 nM T80276 CKJ5C2 58205017 Ki = 1 nM T80276 CVR9Q2 58233988 IC50 = 15.85 nM T80276 CB9AH8 58234990 IC50 = 7000 nM T80276 CJ8YI2 58234995 IC50 = 230 nM T80276 CZF3U5 58235016 IC50 = 200 nM T80276 CM0ND7 58235018 IC50 = 110 nM T80276 C25RXY 58235020 IC50 = 160 nM T80276 CAY94U 58235030 IC50 = 370 nM T80276 CAJC03 58235033 IC50 = 2900 nM T80276 CN7MZ8 58235039 IC50 = 290 nM T80276 CPW84H 58235041 IC50 = 110 nM T80276 C70CRN 58235043 IC50 = 510 nM T80276 C5SQV3 58235052 IC50 = 85 nM T80276 CEZ4T5 58235053 IC50 = 300 nM T80276 C82LIS 58235061 IC50 = 13000 nM T80276 C3SO4E 58235062 IC50 = 90 nM T80276 CZ0SD5 58235073 IC50 = 150 nM T80276 CQP25T 58235077 IC50 = 98 nM T80276 C0LDZ2 58235079 IC50 = 810 nM T80276 C2YG5L 58235088 IC50 = 220 nM T80276 CU3WG8 58298312 IC50 > 30000 nM T80276 C7GIQ1 58298333 IC50 = 6200 nM T80276 CZUO79 58441681 IC50 = 0.1 nM T80276 CB2VP8 58507929 Ki = 27.4 nM T80276 CK0O4B 58508043 Ki = 53.7 nM T80276 C1I4ZO 58508110 Ki = 88.9 nM T80276 C85HOT 58508283 Ki = 8.3 nM T80276 CTEX03 59244213 IC50 = 48 nM T80276 CWL3G4 59244242 IC50 = 2400 nM T80276 CGLV53 59244245 IC50 = 440 nM T80276 CMDX18 59244276 IC50 = 220 nM T80276 CMV67Z 59244308 IC50 > 50000 nM T80276 CO9E4L 59244337 IC50 = 40 nM T80276 C5KEP0 59244360 IC50 = 42 nM T80276 CHLE28 59244510 IC50 = 410 nM T80276 C6JO8I 59244527 IC50 = 120 nM T80276 CG09EI 59244568 IC50 = 32 nM T80276 C9VLB1 59244594 IC50 = 46 nM T80276 CQ7BO0 59244626 IC50 = 1700 nM T80276 C4L7SI 59244670 IC50 = 26 nM T80276 C1CRV9 59244679 IC50 = 35 nM T80276 C25MLK 59244698 IC50 = 14 nM T80276 CF48RM 59244739 IC50 = 200 nM T80276 CLJ09R 59244842 IC50 = 22600 nM T80276 C18ZMW 59244873 IC50 = 3700 nM T80276 C3CX6J 59244888 IC50 = 19000 nM T80276 CMT5B3 59244941 IC50 = 25 nM T80276 CV7K1T 59244961 IC50 > 50000 nM T80276 CJ6R8Q 59251679 IC50 = 3.6 nM T80276 CWKJ69 59251709 IC50 = 13 nM T80276 C0X1KW 59251723 IC50 = 26 nM T80276 CCS6A3 59251739 IC50 = 25 nM T80276 C4WOM8 59251754 IC50 = 2000 nM T80276 C9H6EQ 59251763 IC50 = 36 nM T80276 C81CTW 59251796 IC50 = 16 nM T80276 CXJP65 59251818 EC50 < 40 nM T80276 C42WUB 59251834 IC50 = 2 nM T80276 CGB6E7 59251838 IC50 = 68 nM T80276 CHC07M 59251845 IC50 = 8 nM T80276 CWF9Z7 59251848 IC50 = 33 nM T80276 CV65WP 59251849 IC50 = 260 nM T80276 CVGU78 59251850 IC50 = 11 nM T80276 C3UDA9 59251852 IC50 = 7.9 nM T80276 CN4EA6 59251922 IC50 = 5 nM T80276 C10UAH 59251938 IC50 = 54 nM T80276 CT81MH 59251951 IC50 = 2 nM T80276 CZOJ61 59251964 IC50 = 3 nM T80276 C1G2UV 59251975 EC50 = 60 nM T80276 CB3OZ0 59251984 IC50 = 14 nM T80276 CRZ5B1 59251991 IC50 = 40 nM T80276 C1X8TM 59252012 IC50 = 1200 nM T80276 C2I4WY 59252083 IC50 = 6 nM T80276 C3NKS2 59259019 IC50 = 2.8 nM T80276 CILJ94 59293648 IC50 = 22 nM T80276 C6A3KL 59293676 IC50 = 12 nM T80276 CC14ZL 59293709 IC50 = 19 nM T80276 C0R3TX 59293715 IC50 = 100 nM T80276 C9TVC6 59293721 IC50 = 39 nM T80276 CZ5OV1 59293740 IC50 = 170 nM T80276 CB2Z4R 59293755 IC50 = 9.5 nM T80276 C8AL6C 59293763 IC50 = 440 nM T80276 CTMA05 59453047 IC50 = 510 nM T80276 CYN1L2 59453060 IC50 = 11100 nM T80276 C1I7QA 59453069 IC50 = 120 nM T80276 CNV0I9 59453076 IC50 = 1900 nM T80276 CQYI53 59453077 IC50 = 2500 nM T80276 CV6A4J 59453078 IC50 = 526 nM T80276 CV1SY9 59453083 IC50 = 4700 nM T80276 CPH5N4 59453087 IC50 = 10500 nM T80276 C0WQ4N 59453111 IC50 = 100 nM T80276 CWJ3L7 59453121 IC50 = 200 nM T80276 CLQ08G 59453125 IC50 = 3200 nM T80276 CXA9D8 59453133 IC50 = 3800 nM T80276 CT3CF1 59477024 IC50 > 39810.72 nM T80276 CF6YB8 59477038 IC50 > 100000 nM T80276 CK3H9O 59477041 IC50 = 10000 nM T80276 C7KG5E 59477042 IC50 > 100000 nM T80276 C01DZW 59477048 IC50 > 10000 nM T80276 C5D6ZW 59477194 IC50 = 5300 nM T80276 CTA78B 59507597 IC50 = 2.6 nM T80276 CR9Q3B 59507602 IC50 = 34 nM T80276 C0L9FP 59507663 IC50 = 2.4 nM T80276 CAJ1Y5 59507725 IC50 = 21 nM T80276 C7UMJ8 59507731 IC50 = 7.4 nM T80276 CPB1A4 59507734 IC50 = 4.1 nM T80276 CK09SM 59507757 IC50 = 15 nM T80276 CJG2L3 59507767 IC50 = 14 nM T80276 C1PNB0 59507839 IC50 = 23 nM T80276 CDB14C 59507892 IC50 = 2.2 nM T80276 CH9KB4 59507919 IC50 = 8 nM T80276 C09HWE 59507937 IC50 = 18.4 nM T80276 CY3VA0 59507952 IC50 = 68 nM T80276 C2X8TY 59548177 Ki = 150 nM T80276 C41QVZ 59548192 Ki = 161 nM T80276 CGRO45 59548196 Ki = 270 nM T80276 CD39AG 59548207 Ki > 10000 nM T80276 C6KP4G 59548220 Ki = 200 nM T80276 C8XOU3 59548222 Ki = 114 nM T80276 CTNU85 59548226 Ki = 240 nM T80276 CLB6N4 59548232 Ki = 8300 nM T80276 CSWV07 59548243 Ki = 260 nM T80276 CMT2R0 59548250 Ki = 620 nM T80276 C3I8NE 59548256 Ki = 280 nM T80276 CJXP84 59548260 Ki = 1.9 nM T80276 C8W5HT 59548263 Ki = 640 nM T80276 CT8Q5B 59548274 Ki = 8 nM T80276 CVF1B2 59548283 Ki = 120 nM T80276 CY31EA 59548284 Ki = 280 nM T80276 CO4GT7 59548288 Ki = 7.7 nM T80276 CFR7S8 59548302 Ki = 63 nM T80276 CK4QO7 59548308 Ki = 360 nM T80276 CRM20Z 59548320 Ki = 160 nM T80276 C26MJV 59548335 Ki = 11 nM T80276 CJE5I4 59548341 Ki = 250 nM T80276 C8O1VS 59548349 Ki = 16 nM T80276 CZE96K 59548353 Ki = 43 nM T80276 CWC65A 59548356 Ki = 22 nM T80276 CMKP95 59548371 Ki = 55 nM T80276 CC8UV3 59548383 Ki = 67 nM T80276 CD4ET2 59548402 Ki = 120 nM T80276 CES59T 59548403 Ki = 520 nM T80276 CE8P3G 59548407 Ki = 18 nM T80276 C63PCW 59548408 Ki = 9.7 nM T80276 CO4K2W 59548419 Ki = 9.3 nM T80276 CSDB78 59548424 Ki = 9 nM T80276 C81FCQ 59548431 Ki = 17 nM T80276 CX51UI 59548437 Ki = 13 nM T80276 CQ73ND 59548444 Ki = 16 nM T80276 C0VP1T 59548448 Ki = 16 nM T80276 CLGY34 59548453 Ki = 59 nM T80276 CBT21W 59548454 Ki = 150 nM T80276 CJT68K 59548460 Ki = 290 nM T80276 C9LFT3 59548462 Ki = 3 nM T80276 CJGZ14 59548471 Ki = 11 nM T80276 CX8C2U 59548480 Ki = 3200 nM T80276 CR53FU 59604291 IC50 > 3000 nM T80276 CT7J2V 59604295 IC50 > 10000 nM T80276 C90ZIF 59604376 IC50 = 693 nM T80276 CFKT64 59604403 IC50 > 3000 nM T80276 CEU3P6 59604432 IC50 = 1090 nM T80276 CA2RH5 59604449 IC50 = 1131 nM T80276 CGM80S 59604527 IC50 = 459 nM T80276 CGF48E 59604531 IC50 = 259 nM T80276 CQ31SH 59604532 IC50 = 89 nM T80276 CZ4V7F 59604618 IC50 > 3000 nM T80276 C4OUK8 59604658 IC50 = 2447 nM T80276 C78IGQ 59604689 IC50 = 1092 nM T80276 COLJ98 59604770 IC50 = 763 nM T80276 CQ69DM 59604853 IC50 = 238 nM T80276 C7BPD5 59604870 IC50 = 1048 nM T80276 CLP3G4 59604871 IC50 = 2344 nM T80276 C5XU7F 59604897 IC50 = 670 nM T80276 CX34TW 59604899 IC50 = 2895 nM T80276 CCK78R 59604980 IC50 > 3000 nM T80276 CE89OV 59605039 IC50 = 1800 nM T80276 CYL9G0 59605041 IC50 = 2172 nM T80276 CR1Y9N 59605098 IC50 > 3000 nM T80276 C2QZ8T 59605139 IC50 = 137 nM T80276 C5VP8F 59605730 Ki = 236 nM T80276 CHO01A 59606100 Ki = 110 nM T80276 CW9VH5 59606123 Ki = 157 nM T80276 C4Y3GL 59609976 IC50 = 85 nM T80276 C1PC0J 59634638 IC50 > 20000 nM T80276 CP2UY3 59634686 IC50 = 17600 nM T80276 C1TH2N 59634692 IC50 = 4400 nM T80276 CPA0L2 59634709 IC50 = 16800 nM T80276 CBI0M6 59688563 IC50 = 125.89 nM T80276 COFZ83 59753763 IC50 = 2200 nM T80276 CUYB59 60148924 IC50 = 6600 nM T80276 CM8PD7 60150509 IC50 = 1600 nM T80276 C5KD3Z 60154714 Ki > 10000 nM T80276 CS0L4D 60154996 Ki > 10000 nM T80276 C1UI3P 60155086 Ki = 4900 nM T80276 CX08ON 60155087 Ki = 1300 nM T80276 CX8J1I 60155265 Ki = 49 nM T80276 CAT40I 60155266 Ki = 22 nM T80276 CD56VA 60155268 Ki = 39 nM T80276 CCQB56 60155375 IC50 = 38 nM T80276 CH5X2S 60155376 IC50 = 220 nM T80276 C74FEN 60155377 IC50 = 744 nM T80276 CZ6G4B 60155378 IC50 = 174 nM T80276 C10AHQ 60155379 IC50 = 142 nM T80276 C5FI4P 60155451 Ki = 94 nM T80276 CX9G4U 60155452 Ki = 84 nM T80276 C9Q7DE 60155469 IC50 = 97 nM T80276 CH8UY5 60155470 IC50 = 752 nM T80276 C3EDY4 60155471 IC50 = 1807 nM T80276 CE0ZX1 60155472 IC50 = 953 nM T80276 CG90MC 60155473 IC50 = 200 nM T80276 C82PVI 60155474 IC50 = 3643 nM T80276 CX49FT 60155475 IC50 = 3381 nM T80276 CR7EG9 60155538 Ki = 33 nM T80276 CU6YB9 60155539 Ki = 73 nM T80276 CW6N1S 60155552 IC50 = 90 nM T80276 CIB08V 60155553 IC50 = 323 nM T80276 CZE28G 60155554 IC50 = 316 nM T80276 CZD2W7 60155555 IC50 = 290 nM T80276 CO6IU3 60155556 IC50 = 727 nM T80276 C6HN5O 60155557 IC50 = 174 nM T80276 CMQ9G1 60155638 IC50 = 476 nM T80276 CG56KT 60155639 IC50 = 142 nM T80276 CBJ65P 60155640 IC50 = 705 nM T80276 C8OJK0 60155641 IC50 = 209 nM T80276 CT9XJ6 60155642 IC50 = 972 nM T80276 C5BYQ3 60155643 IC50 = 323 nM T80276 C57RBF 60155722 IC50 = 555 nM T80276 CU7J6L 60155723 IC50 = 2369 nM T80276 CSZA16 60155724 IC50 = 342 nM T80276 C21DWT 60155725 IC50 = 4647 nM T80276 C12CQU 60155726 IC50 = 1663 nM T80276 CA5TM3 60155805 IC50 = 234 nM T80276 C60RIO 60155806 IC50 = 110 nM T80276 CKWI93 60155892 IC50 > 10000 nM T80276 C3EK2G 60155994 IC50 > 10000 nM T80276 C54INX 60161770 IC50 = 10000 nM T80276 CX6NA3 60161903 IC50 > 10000 nM T80276 CB59LY 60161905 IC50 = 80 nM T80276 CTZW84 60161907 IC50 > 20000 nM T80276 CU87AK 60162043 IC50 = 740 nM T80276 C1EWV9 60162169 IC50 = 800 nM T80276 CQC25X 60162301 IC50 = 600 nM T80276 C04WJY 60163476 IC50 = 60 nM T80276 CV0MD4 62705168 Ki = 1450 nM T80276 CSD3F8 62705169 Ki = 1270 nM T80276 C3LS8Q 62705170 Ki > 4550 nM T80276 C2E3AO 62705171 Ki > 4550 nM T80276 CSD0N6 62705990 IC50 = 648 nM T80276 C9NI6K 62705991 IC50 = 654 nM T80276 C2RDA4 62706154 IC50 = 306 nM T80276 C3M6QC 62706155 IC50 = 119 nM T80276 CAG23H 62706156 IC50 = 120 nM T80276 C1RB8F 62706157 IC50 = 393 nM T80276 CGC62F 62706158 IC50 = 73 nM T80276 C67TAB 62706159 IC50 = 268 nM T80276 C4IGR0 62706312 IC50 = 239 nM T80276 CPM5R9 62706313 IC50 = 85 nM T80276 CX6IU3 62706314 IC50 = 68 nM T80276 CFJ8W5 62706315 IC50 = 96 nM T80276 CX0H7E 62706316 IC50 = 463 nM T80276 C06IUA 62706317 IC50 = 144 nM T80276 C82NPI 62706470 IC50 = 177 nM T80276 CPR50J 62706471 IC50 = 635 nM T80276 CA31ZB 62706472 IC50 = 5840 nM T80276 CWRJ86 62706475 IC50 = 1140 nM T80276 CNMX21 62706476 IC50 = 3020 nM T80276 CS0CA6 62706650 IC50 = 47 nM T80276 C71APZ 62706651 IC50 = 122 nM T80276 CFBD83 62706652 IC50 = 1140 nM T80276 CL20FV 62706653 IC50 = 173 nM T80276 C34MPU 62706654 IC50 = 105 nM T80276 CHX01T 62706655 IC50 = 1660 nM T80276 CM39TP 62706813 IC50 = 112 nM T80276 CHK4I1 62706814 IC50 = 4580 nM T80276 C16ZGX 62706815 IC50 = 4290 nM T80276 CS4VA8 62706816 IC50 > 125000 nM T80276 CY0D8M 62706817 IC50 = 3170 nM T80276 C9G5NA 62707451 Ki = 514 nM T80276 CWZ1I7 62707452 Ki > 4550 nM T80276 C80KUA 62707599 Ki = 3000 nM T80276 CIRO73 66493714 IC50 = 552 nM T80276 C71LPV 66493729 IC50 = 914 nM T80276 CU21FZ 66546792 IC50 = 27 nM T80276 C54NOW 66552297 IC50 > 100000 nM T80276 CX4HW1 66552298 IC50 > 100000 nM T80276 CEJ54A 66552343 IC50 > 100000 nM T80276 CUQ5Y2 66552345 IC50 > 19952.62 nM T80276 C5F8ZE 66552346 IC50 > 100000 nM T80276 CHQC56 66552347 IC50 > 100000 nM T80276 CS6BQ0 66552348 IC50 = 6309.57 nM T80276 CGT2V9 66552407 IC50 > 63095.73 nM T80276 CIJ3C5 66552408 IC50 > 3162.28 nM T80276 C6ZFI1 66552410 IC50 > 100000 nM T80276 C8S7CM 66552411 IC50 > 3981.07 nM T80276 C9A7IK 66552412 IC50 > 100000 nM T80276 CRC24S 66552467 IC50 > 100000 nM T80276 CHU5V3 66552468 IC50 > 100000 nM T80276 C46POH 66552523 IC50 > 100000 nM T80276 C68LXT 66552524 IC50 > 100000 nM T80276 C91JZL 66553214 IC50 > 10000 nM T80276 CUC7B3 66557964 IC50 = 13 nM T80276 C9X2TB 66558056 IC50 = 19 nM T80276 C1R3SI 66653673 IC50 = 6190 nM T80276 CF8BZ7 66677439 IC50 = 2150 nM T80276 C0X9FR 66699750 IC50 = 1380 nM T80276 CN0RE8 66779813 IC50 = 2000 nM T80276 C3IP5D 66779815 IC50 = 1300 nM T80276 CH86MR 66779905 IC50 = 4000 nM T80276 CX2N6E 66779920 IC50 > 3200 nM T80276 C9O4TC 66779989 IC50 = 1600 nM T80276 CF2UM8 66780001 IC50 > 3200 nM T80276 CHU0C5 66780007 IC50 = 250 nM T80276 CGL4V1 66780016 IC50 = 2500 nM T80276 C5F6OA 66780027 IC50 = 7900 nM T80276 C8DN7A 66780034 IC50 = 3200 nM T80276 C4AM6R 66780100 IC50 > 4000 nM T80276 CZ5P2N 66780118 IC50 = 400 nM T80276 CREA54 66780266 IC50 = 1000 nM T80276 CRCA72 66780292 IC50 = 2000 nM T80276 CW2SM6 66780337 IC50 = 500 nM T80276 CU54DY 66780379 IC50 = 2500 nM T80276 CQ70YA 66780434 IC50 > 2500 nM T80276 C8F9UY 66780515 IC50 = 630 nM T80276 CFH6C2 66780644 IC50 = 2500 nM T80276 CTZB46 66780835 IC50 = 2500 nM T80276 CEP5A2 66780844 IC50 = 50000 nM T80276 CB8WP9 66788776 Ki = 8.3 nM T80276 C51ARE 66788835 IC50 = 4.5 nM T80276 C6DYG9 66788911 Ki = 6.5 nM T80276 CQ5TC4 66789238 Ki = 43 nM T80276 CIR86Z 66789609 Ki = 148 nM T80276 CYKD92 66789704 Ki = 26 nM T80276 CRO34N 66790135 Ki = 6.1 nM T80276 COE7X1 66790311 Ki = 54 nM T80276 CUJB72 66790335 Ki = 5.7 nM T80276 CW12XO 66882257 IC50 > 10000 nM T80276 C6IO1S 66883557 IC50 > 10000 nM T80276 C1HSE0 67035086 IC50 = 1400 nM T80276 C38RGB 67035556 IC50 > 9000 nM T80276 CV3HW2 67035568 IC50 > 9000 nM T80276 C8HOZ9 67041250 IC50 = 5500 nM T80276 C5E4AJ 67050504 IC50 = 14 nM T80276 CMWO25 67061712 Ki = 0.14 nM T80276 CU58AM 67073110 Ki = 0.35 nM T80276 C1K5PQ 67094257 Ki = 380 nM T80276 CJ46YU 67094333 Ki = 370 nM T80276 C0OX5N 67103709 IC50 = 140 nM T80276 C9J2EO 67103712 IC50 = 25 nM T80276 CM4W1Y 67103722 IC50 = 170 nM T80276 C5TYQ3 67103909 IC50 = 12 nM T80276 CVJ49E 67103974 IC50 = 180 nM T80276 C3VFY7 67104025 IC50 = 3000 nM T80276 CC07KA 67104052 IC50 = 2600 nM T80276 C7EZW6 67192973 IC50 = 370 nM T80276 CQHF85 67284779 IC50 = 3960 nM T80276 CT6BX3 67285457 Ki > 125000 nM T80276 C1HBC0 67535197 IC50 = 18 nM T80276 CNZ2C3 67535447 Ki = 529 nM T80276 C3M1OJ 67535551 Ki = 5.6 nM T80276 C25AHY 67984037 IC50 = 6200 nM T80276 C97SXL 68194826 IC50 = 31.62 nM T80276 C8I7GC 68293638 IC50 > 10000 nM T80276 CX1HO4 68295238 IC50 = 1600 nM T80276 C62YGS 68295435 IC50 > 20000 nM T80276 CMG58Q 68295585 IC50 = 60 nM T80276 CIU6P5 68295624 IC50 > 20000 nM T80276 CYZ6P3 68313479 IC50 = 3.6 nM T80276 CVRP38 68353609 IC50 = 49 nM T80276 CP4UF3 68353647 IC50 = 140 nM T80276 CI1HJ5 68504925 IC50 > 1000 nM T80276 C01QHM 68547896 IC50 = 400 nM T80276 CB03UO 68774589 IC50 = 705 nM T80276 C45TIJ 69489467 IC50 = 15.4 nM T80276 C0L9EF 70675845 IC50 > 83300 nM T80276 CN09DI 70675846 IC50 = 27200 nM T80276 CNX20F 70676303 Ki = 2 nM T80276 CH7PL5 70681202 Ki = 3 nM T80276 C6BQE1 70681248 IC50 = 2500 nM T80276 CPE36T 70681262 IC50 = 1300 nM T80276 C3F6OC 70681276 IC50 = 21830 nM T80276 CPX41V 70682086 IC50 = 1258.93 nM T80276 CDMO03 70682114 IC50 = 2.7 nM T80276 CQW54O 70682591 Ki = 200 nM T80276 CPV59G 70682592 Ki = 20 nM T80276 CZ6XC8 70682805 IC50 = 4100 nM T80276 CCGB61 70683291 Ki = 13 nM T80276 CB3ZN5 70683337 IC50 = 2500 nM T80276 C1I5PH 70683338 IC50 = 320 nM T80276 CSM0A6 70684204 IC50 = 794.33 nM T80276 C65LPD 70684413 Ki > 4550 nM T80276 CXD08N 70684690 Ki = 28 nM T80276 CG95EC 70684794 Ki = 1.73 nM T80276 C8O2QH 70685440 IC50 = 630 nM T80276 CZG9M1 70685441 IC50 = 400 nM T80276 CH7KO0 70685442 IC50 = 320 nM T80276 CM3R0C 70685462 IC50 = 79 nM T80276 C6G4WB 70686339 IC50 > 100000 nM T80276 CON8X4 70686340 IC50 > 19952.62 nM T80276 C1ASW4 70686341 IC50 = 1995.26 nM T80276 CP10AJ 70686372 IC50 = 35.1 nM T80276 C0PWL5 70686455 IC50 > 5011.87 nM T80276 CN4CR2 70686584 IC50 = 2600 nM T80276 C85FWA 70686829 Ki = 30 nM T80276 CQS8G7 70686830 Ki = 5 nM T80276 C8QSD2 70688455 IC50 = 794.33 nM T80276 CMC74I 70688479 IC50 = 34.3 nM T80276 CFCJ02 70688558 IC50 = 1258.93 nM T80276 CSX6I7 70688908 Ki = 110 nM T80276 C1U5FC 70689024 IC50 = 120 nM T80276 CJ61UF 70689026 IC50 = 480 nM T80276 CQ04ZJ 70689027 IC50 = 8.1 nM T80276 C0XF8W 70689122 IC50 = 2200 nM T80276 C5YN6U 70689166 IC50 > 4000 nM T80276 CCBS90 70689600 Ki = 175 nM T80276 C6L4WY 70689639 IC50 = 630 nM T80276 CL9BF7 70689663 IC50 > 50000 nM T80276 CGT1X2 70690496 IC50 = 630.96 nM T80276 CN45VU 70690535 IC50 = 30.3 nM T80276 CW3U5J 70690994 Ki = 190 nM T80276 CCGA03 70691211 IC50 > 10000 nM T80276 CC6I1Q 70691259 IC50 > 2000 nM T80276 C0Z9PM 70691729 Ki = 1280 nM T80276 CD3JL4 70691776 IC50 = 1600 nM T80276 C1BOP6 70691801 IC50 = 440 nM T80276 CC64RD 70692128 IC50 > 300000 nM T80276 C7ASK8 70692129 IC50 > 48000 nM T80276 CDK52M 70692650 IC50 > 15848.93 nM T80276 CGQJ68 70692914 IC50 > 100 nM T80276 C7G5UV 70692915 IC50 > 100 nM T80276 C3TM1F 70693128 Ki = 35 nM T80276 C2VAU8 70693129 Ki = 11 nM T80276 CU3WF2 70693248 IC50 = 10.2 nM T80276 C4SEX0 70693329 IC50 = 295 nM T80276 CWY7O2 70693330 IC50 = 5200 nM T80276 C4P9CL 70693798 Ki = 1.7 nM T80276 CJ76QG 70693799 Ki = 1.8 nM T80276 CX2JZ1 70694178 IC50 > 24000 nM T80276 C7HW2B 70694179 IC50 > 100000 nM T80276 CICE82 70694721 IC50 = 0.6 nM T80276 C38LWS 70694722 IC50 = 26 nM T80276 C65FHO 70694723 Ki = 1.9 nM T80276 CPFO83 70694805 IC50 > 5011.87 nM T80276 CRNY76 70695188 Ki = 45 nM T80276 C3N5YJ 70695189 Ki = 187 nM T80276 CQM5N7 70695335 IC50 = 98.5 nM T80276 CLY5G3 70695401 IC50 = 2350 nM T80276 C75YGN 70695469 IC50 = 2000 nM T80276 C7KIH1 70695983 IC50 = 25 nM T80276 C61CFG 70696737 IC50 > 3162.28 nM T80276 C7KL5X 70696852 IC50 > 25118.86 nM T80276 C1A3MP 70697347 IC50 = 244 nM T80276 CCG28A 70697442 IC50 > 10000 nM T80276 CF8EK2 71250848 IC50 = 2600 nM T80276 CJP69K 71250855 IC50 > 10000 nM T80276 C8KD6L 71250859 IC50 > 10000 nM T80276 CM10HY 71250872 IC50 = 1300 nM T80276 CS3V1R 71250875 IC50 > 10000 nM T80276 C85IZO 71250882 IC50 = 3200 nM T80276 C1LI6X 71250891 IC50 = 400 nM T80276 CSO29K 71250896 IC50 > 10000 nM T80276 CKE7H2 71250907 IC50 > 10000 nM T80276 CI5MT1 71250909 IC50 > 10000 nM T80276 C9G2MT 71250929 IC50 = 3000 nM T80276 CZP1E8 71250935 IC50 > 10000 nM T80276 CRH8E2 71270723 IC50 = 158.49 nM T80276 CWR58A 71270783 IC50 > 1995.26 nM T80276 CF9LU4 71270807 IC50 = 316.23 nM T80276 C7FDL2 71270817 IC50 = 199.53 nM T80276 CNR1G9 71270824 IC50 > 1584.89 nM T80276 C38LBA 71270831 IC50 = 316.23 nM T80276 CTL6R5 71270836 IC50 = 158.49 nM T80276 CM4LX7 71270848 IC50 > 6309.57 nM T80276 C2GWX6 71270906 IC50 > 1584.89 nM T80276 CX0DL3 71270910 IC50 = 1584.89 nM T80276 C0COW6 71270913 IC50 > 6309.57 nM T80276 CB0S8G 71270927 IC50 = 199.53 nM T80276 C24IOW 71270948 IC50 > 1995.26 nM T80276 C5BJ2Y 71270957 IC50 > 1000 nM T80276 C03NFY 71271625 IC50 > 5011.87 nM T80276 CL47JU 71271739 IC50 > 1584.89 nM T80276 CS5JG6 71271910 IC50 = 2511.89 nM T80276 C4PSK8 71271965 IC50 = 501.19 nM T80276 CB4N1M 71272066 IC50 > 1995.26 nM T80276 CD8E1Y 71272453 IC50 = 316.23 nM T80276 C8EW9V 71272757 IC50 = 251.19 nM T80276 C0LO8I 71272765 IC50 = 630.96 nM T80276 C42PJQ 71449564 IC50 > 83300 nM T80276 CFN52U 71449565 IC50 = 100000 nM T80276 CK58RV 71449587 IC50 = 44 nM T80276 C7ULC4 71449776 IC50 = 51500 nM T80276 CTL30H 71450452 IC50 = 195 nM T80276 CH9ZB4 71450646 Ki = 3.5 nM T80276 CWQF08 71450647 Ki = 13 nM T80276 CNHJ63 71451228 IC50 = 3575 nM T80276 CLZO91 71451372 IC50 = 52800 nM T80276 CSB2E6 71451587 IC50 = 30800 nM T80276 C9O5HM 71451588 IC50 > 83300 nM T80276 C9SC2V 71452282 IC50 = 112 nM T80276 C7Z6SV 71452476 Ki = 29 nM T80276 C71JEC 71453177 IC50 = 240000 nM T80276 C6VF7J 71453206 IC50 = 43 nM T80276 CR84JX 71453419 Ki = 2 nM T80276 CEKG39 71453424 IC50 = 56900 nM T80276 CF1B5X 71453425 IC50 = 205000 nM T80276 CZ61FJ 71454160 IC50 = 12589254.12 nM T80276 CZ8Q5P 71454238 Ki = 20 nM T80276 C4NS8G 71454916 IC50 = 142000 nM T80276 CIK32W 71454917 IC50 > 83300 nM T80276 CF74SL 71454944 IC50 = 130 nM T80276 CC46RH 71455124 IC50 = 112000 nM T80276 CCP3M4 71455125 IC50 > 83300 nM T80276 CT32GB 71455818 IC50 = 43 nM T80276 CE1IX7 71456728 IC50 = 78 nM T80276 CLUR84 71457607 IC50 = 328 nM T80276 CCPV51 71458543 IC50 > 83300 nM T80276 CMZA06 71458544 IC50 = 41400 nM T80276 CF42GC 71458545 IC50 = 146000 nM T80276 CM1ND2 71458573 IC50 = 80 nM T80276 C3S0NP 71458574 IC50 = 61 nM T80276 CY6WI2 71458575 IC50 = 92 nM T80276 CD50NR 71458791 IC50 = 349000 nM T80276 C1Y8WD 71459503 IC50 = 102 nM T80276 CT7K3A 71460422 IC50 = 33 nM T80276 C8ELG4 71460604 IC50 = 82800 nM T80276 CS7VI3 71460605 IC50 = 76000 nM T80276 CA7QI2 71460606 IC50 = 73700 nM T80276 C1O2ET 71460607 IC50 = 149000 nM T80276 CW9YM2 71461240 IC50 = 46 nM T80276 C2HOB7 71461243 IC50 = 15 nM T80276 CE9I8U 71461426 Ki = 8.6 nM T80276 CRL29X 71461427 Ki = 311 nM T80276 CVQ26M 71462083 IC50 = 119000 nM T80276 CXLQ15 71462308 IC50 = 212000 nM T80276 CZC93M 71463157 Ki = 11 nM T80276 CY74CX 71472903 IC50 = 1530 nM T80276 CB78IN 71493938 IC50 > 10000 nM T80276 CU3EO6 71520393 IC50 = 375 nM T80276 CYC6S1 71520394 IC50 = 9200 nM T80276 C1KMX0 71520395 IC50 = 823 nM T80276 CYK7N8 71520396 IC50 > 10000 nM T80276 CTC0O8 71520397 IC50 = 1050 nM T80276 CHV20S 71520675 IC50 > 50000 nM T80276 C9O0MG 71520767 IC50 > 50000 nM T80276 CCQ4T5 71520768 IC50 > 50000 nM T80276 C63RAI 71520769 IC50 > 50000 nM T80276 CZK53W 71520770 IC50 > 50000 nM T80276 CEZ67P 71520868 IC50 > 50000 nM T80276 C0UZ3D 71526877 IC50 = 3700 nM T80276 CP05SQ 71526878 IC50 = 8100 nM T80276 CZK6X9 71526879 IC50 > 10000 nM T80276 C8QRE4 71526880 IC50 = 2800 nM T80276 CT3QI8 71526881 IC50 = 3300 nM T80276 CO4MY1 71527005 IC50 = 2200 nM T80276 CJC64F 71527006 IC50 = 2300 nM T80276 C96WZG 71527007 IC50 = 720 nM T80276 CUC7I1 71527008 IC50 = 1500 nM T80276 C09WKC 71527009 IC50 = 1600 nM T80276 CSPO76 71527716 IC50 > 5011.87 nM T80276 CIN7O1 71527842 IC50 > 1584.89 nM T80276 CO6CI7 71528725 IC50 = 1500 nM T80276 C5U2ZC 71528726 IC50 = 42 nM T80276 CTKO36 71528727 IC50 = 2300 nM T80276 C2KF3X 71533728 IC50 = 2000 nM T80276 CI7Q4K 71548718 IC50 = 418 nM T80276 CED62L 71548719 IC50 = 283 nM T80276 C4B0KN 71549093 IC50 = 10000 nM T80276 CQ16UM 71584055 IC50 = 1600 nM T80276 C1ZNG7 71600385 IC50 = 398 nM T80276 C1CO2S 71600386 IC50 = 1463 nM T80276 C5IM3B 71600530 IC50 = 2305 nM T80276 CNO5F0 71600792 IC50 > 10000 nM T80276 C10XMI 71600793 IC50 = 3128 nM T80276 C6PRV1 71655831 IC50 = 270 nM T80276 CWG8M3 71682651 IC50 = 20 nM T80276 C6UGW3 71682652 IC50 = 2700 nM T80276 C7BX4K 71682653 IC50 = 620 nM T80276 CQX8N3 71682654 IC50 > 9100 nM T80276 CCG6J1 71682807 IC50 = 320 nM T80276 CS32HB 71716798 IC50 > 1584.89 nM T80276 C07GCV 71716799 IC50 > 1584.89 nM T80276 C9S0BX 71716809 IC50 > 2000 nM T80276 CH8R6V 71717423 IC50 = 885 nM T80276 CFW01E 71718034 IC50 = 431 nM T80276 C1YR0E 71813981 IC50 = 110 nM T80276 CBL68S 71813982 IC50 = 790 nM T80276 C9FA3Y 71813983 IC50 = 1600 nM T80276 CR0UF8 71813984 IC50 = 3800 nM T80276 CIE95Q 71814140 IC50 = 4000 nM T80276 C7EY1Q 72163951 Ki = 190 nM T80276 CVT76M 72163952 Ki = 390 nM T80276 C9UOH5 72164062 Ki > 10000 nM T80276 CT3X8G 72164184 Ki > 10000 nM T80276 C4NE0C 72376504 IC50 = 20.6 nM T80276 CNX76A 72544842 IC50 = 1995.26 nM T80276 C29KOU 72709209 IC50 > 10000 nM T80276 CT73IW 72709284 IC50 = 2700 nM T80276 CIBU31 72792686 IC50 > 10000 nM T80276 CG3N9F 72947195 IC50 = 0.87 nM T80276 CFG97I 72950095 IC50 = 60 nM T80276 C6Q7FI 73052343 IC50 = 2.1 nM T80276 CP7HF0 73345848 IC50 = 2900 nM T80276 C9B3DF 73351941 IC50 = 426 nM T80276 CL0XZ1 73659199 Ki = 132 nM T80276 C8EI1X 73673707 IC50 = 1.3 nM T80276 CBYN18 73977439 IC50 = 3981 nM T80276 C9V1YR 73977449 IC50 = 631 nM T80276 CXA90D 73977451 IC50 = 501 nM T80276 CEZ7L2 73977461 IC50 = 398 nM T80276 CNLT94 74538916 IC50 = 1.1 nM T80276 C5EH2O 74538978 IC50 = 1.5 nM T80276 CF9TU6 74538980 IC50 = 1.6 nM T80276 C8YX6V 74538981 IC50 = 1.1 nM T80276 CW9RX8 74538982 IC50 = 2.1 nM T80276 CIJ91K 74539042 IC50 = 0.75 nM T80276 CE8M6L 74539043 IC50 = 4.8 nM T80276 CWV39P 74539044 IC50 = 0.73 nM T80276 C6Z2XJ 74539045 IC50 = 0.91 nM T80276 CFG83U 74539108 IC50 = 0.82 nM T80276 C2K4NM 74539109 IC50 = 1 nM T80276 CE7RT1 74539682 IC50 > 100 nM T80276 CE83ZS 74539683 IC50 = 1.4 nM T80276 CBP56K 74539744 IC50 = 2.3 nM T80276 CGE38X 74539745 IC50 = 1.1 nM T80276 CAN9P2 74539746 IC50 = 4.5 nM T80276 CD0T9V 74539799 IC50 = 0.65 nM T80276 C1BD5P 74539801 IC50 = 1.4 nM T80276 CA5H8W 74539860 IC50 = 1.2 nM T80276 C17SMG 74539861 IC50 = 1.1 nM T80276 C16KOS 74539862 IC50 = 0.59 nM T80276 CZBS60 74539863 IC50 = 1.7 nM T80276 C96PXY 74539919 IC50 = 1.2 nM T80276 C2B8ID 74539920 IC50 = 1.3 nM T80276 CC3R4K 74539921 IC50 = 1.6 nM T80276 CYO4H5 74539922 IC50 = 1.3 nM T80276 CVGX56 76285477 IC50 = 53.4 nM T80276 CN2MI8 76310247 IC50 > 50000 nM T80276 CKO41J 76310248 IC50 = 106 nM T80276 CEN9Q5 76310249 IC50 = 268 nM T80276 CJCF67 76310250 IC50 = 58 nM T80276 CUI09Y 76310253 IC50 > 10000 nM T80276 CMVX74 76310254 IC50 > 10000 nM T80276 CBI09O 76310352 IC50 = 31.16 nM T80276 CMF0R5 76310353 IC50 = 9.9 nM T80276 C06OME 76310354 IC50 = 23.14 nM T80276 CIBQ59 76311315 IC50 = 2130 nM T80276 C8BD3K 76311316 IC50 = 240 nM T80276 C6F1CR 76311317 IC50 = 720 nM T80276 C7IDU0 76311318 IC50 = 2470 nM T80276 CG40TB 76311319 IC50 > 1000 nM T80276 C5WSZ8 76311320 IC50 > 1000 nM T80276 C0M5SE 76311321 IC50 > 1000 nM T80276 CA2VR6 76311340 IC50 = 615 nM T80276 CMR07I 76313939 IC50 = 29400 nM T80276 C5P2CJ 76313940 IC50 = 6970 nM T80276 CAV5Q9 76313941 IC50 = 5800 nM T80276 C4BT9H 76314027 IC50 = 42.84 nM T80276 CC8NB4 76314028 IC50 = 35.6 nM T80276 CCY5L6 76314906 IC50 > 1000 nM T80276 CE3Z1I 76314907 IC50 > 1000 nM T80276 CFY10G 76314908 IC50 = 1280 nM T80276 C4UHR5 76314909 IC50 = 4030 nM T80276 C1B3VO 76314910 IC50 > 1000 nM T80276 CY0Z4U 76314911 IC50 > 1000 nM T80276 CTVO82 76314912 IC50 > 1000 nM T80276 CCWP56 76314913 IC50 = 3000 nM T80276 CO13XZ 76314937 IC50 = 953 nM T80276 C7W2HI 76314938 IC50 = 894 nM T80276 C6H9EL 76314939 IC50 = 591 nM T80276 C0J6PL 76317466 IC50 > 50000 nM T80276 CVW35P 76317467 IC50 > 50000 nM T80276 CZ1T3C 76317468 IC50 = 11920 nM T80276 C4MKN3 76317469 IC50 = 40 nM T80276 C3JA4F 76317470 IC50 = 171 nM T80276 C4XJ5Y 76317471 IC50 = 317 nM T80276 CDTO72 76317570 IC50 = 39.65 nM T80276 C3XYV1 76317571 IC50 = 2.45 nM T80276 CPK6B4 76317572 IC50 = 174.28 nM T80276 C3SIE7 76318525 IC50 = 1260 nM T80276 CU6G7L 76318526 IC50 > 1000 nM T80276 CC3Z2U 76318527 IC50 = 370 nM T80276 CS6ME5 76318566 IC50 = 738 nM T80276 CG4I2R 76318567 IC50 = 625 nM T80276 C8E4GI 76321204 IC50 = 61 nM T80276 CF4OI8 76321205 IC50 = 1400 nM T80276 COW61Q 76321207 IC50 > 10000 nM T80276 CLI04Y 76321208 IC50 = 40.9 nM T80276 CPLO52 76321296 IC50 = 8.6 nM T80276 CGY1N5 76321297 IC50 > 10000 nM T80276 C34OYK 76321298 IC50 = 2 nM T80276 CE35LN 76321299 IC50 = 6.45 nM T80276 CR61ZP 76322185 IC50 > 1000 nM T80276 C5LT0B 76322186 IC50 > 1000 nM T80276 C19SKA 76322187 IC50 > 1000 nM T80276 C1YFK9 76322218 IC50 = 772 nM T80276 CL0T7B 76322219 IC50 = 341 nM T80276 CDG8V4 76324821 IC50 = 27 nM T80276 CJW39V 76324822 IC50 > 50000 nM T80276 C2BFA1 76324823 IC50 = 144 nM T80276 CZTR31 76324910 IC50 = 72.59 nM T80276 C4FMR8 76324911 IC50 = 60.51 nM T80276 CVUB96 76324912 IC50 = 37.33 nM T80276 C8X9TV 76324913 IC50 = 35.41 nM T80276 C1HFI9 76325446 IC50 = 1319 nM T80276 C7IFD5 76325803 IC50 > 1000 nM T80276 C2NK4S 76325804 IC50 > 1000 nM T80276 COJ6P9 76325805 IC50 > 1000 nM T80276 C2AJ6T 76325806 IC50 = 590 nM T80276 C4GZ1Q 76325833 IC50 > 1000 nM T80276 CQ31CA 76325834 IC50 = 792 nM T80276 C4A8XZ 76328376 IC50 = 555 nM T80276 CUQJ87 76328381 IC50 = 1210 nM T80276 CX3N7R 76328473 IC50 = 3.43 nM T80276 CE5I7T 76328474 IC50 = 13.6 nM T80276 CUC04I 76328475 IC50 = 69.11 nM T80276 C8S2IL 76329389 IC50 > 1000 nM T80276 CAEW42 76329390 IC50 > 1000 nM T80276 CMC32D 76329391 IC50 > 1000 nM T80276 CAZ9Q2 76329392 IC50 > 1000 nM T80276 C06ZQJ 76329393 IC50 = 140 nM T80276 C39CLE 76329428 IC50 = 679 nM T80276 CYR0G6 76332050 IC50 = 2500 nM T80276 C4MID5 76332051 IC50 = 1360 nM T80276 C70WJE 76332052 IC50 = 45 nM T80276 CRA39N 76332054 IC50 = 990 nM T80276 CKD7H2 76332159 IC50 = 5551 nM T80276 C8SL3V 76332160 IC50 = 15.2 nM T80276 C3KIG0 76332161 IC50 = 12.03 nM T80276 CE6BI0 76332666 IC50 = 395 nM T80276 CKG1E0 76333034 IC50 = 300 nM T80276 C6D4RU 76333035 IC50 > 1000 nM T80276 CSAT72 76333036 IC50 > 1000 nM T80276 C1JRO2 76333037 IC50 > 1000 nM T80276 C8TNI0 76333038 IC50 > 1000 nM T80276 C16SRX 76333068 IC50 = 527 nM T80276 CW81MC 76333069 IC50 = 946 nM T80276 C26CKL 76333070 IC50 = 503 nM T80276 C47NLT 76333071 IC50 = 836 nM T80276 CZ92PW 76335665 IC50 = 59 nM T80276 C69ATM 76335666 IC50 = 31800 nM T80276 C0SI4C 76335667 IC50 > 50000 nM T80276 C31NEK 76335668 IC50 = 1400 nM T80276 CL6BV5 76335669 IC50 > 50000 nM T80276 C73KJD 76335670 IC50 = 92 nM T80276 CD2KU1 76335780 IC50 = 174.88 nM T80276 C47ZNT 76335781 IC50 = 5.95 nM T80276 CSCK18 76335782 IC50 = 2.9 nM T80276 CRD94L 76335783 IC50 = 6 nM T80276 C6VCF1 76335784 IC50 = 2.42 nM T80276 CT1UL6 76335785 IC50 = 116.75 nM T80276 CU86DF 76335786 IC50 = 14.27 nM T80276 CP2UC5 76336660 IC50 > 1000 nM T80276 C79JAI 76336661 IC50 = 170 nM T80276 CJ3V6Y 76336695 IC50 = 813 nM T80276 CD03GB 76336696 IC50 = 851 nM T80276 C04SRC 77147259 IC50 = 356 nM T80276 C9I7TY 78319187 IC50 = 6309.57 nM T80276 C24LQH 78320362 IC50 = 1300 nM T80276 C9T8KF 78320671 IC50 = 5208 nM T80276 CI2YN8 78320672 IC50 = 393 nM T80276 CI6K4J 78320673 IC50 = 3700 nM T80276 COFJ16 78320996 IC50 > 10000 nM T80276 CMU5P2 78321310 IC50 = 7700 nM T80276 CE13AJ 78321314 IC50 = 1600 nM T80276 CSP2H4 78321635 IC50 = 4700 nM T80276 CWA0B1 78322567 IC50 = 2800 nM T80276 CH6P9D 78322877 IC50 > 10000 nM T80276 C4IW9V 78323193 IC50 = 3100 nM T80276 CD1JC8 78324443 IC50 = 2340 nM T80276 C0V8OG 86306050 IC50 > 10000 nM T80276 C37LKW 86346018 IC50 = 920 nM T80276 C5P3RO 86647783 IC50 = 210 nM T80276 CDXM47 86677874 IC50 > 20000 nM T80276 CP3W1B 86695297 IC50 > 20000 nM T80276 CA17UE 86732669 IC50 = 262 nM T80276 CI8X3C 87150169 IC50 = 3162.28 nM T80276 CV6PI8 87562294 IC50 = 251.19 nM T80276 CEQ80V 89034380 Ki = 20 nM T80276 C1HB3F 89051931 IC50 = 24 nM T80276 CTE1L0 89517065 IC50 = 79 nM T80276 C56KSC 89517226 IC50 = 462 nM T80276 CI1PQ9 89896458 IC50 = 540 nM T80276 CC4SY6 89896459 IC50 = 730 nM T80276 C2VQC1 89896555 IC50 = 200 nM T80276 CP7XG5 89903188 IC50 = 400 nM T80276 CI54WQ 89996408 IC50 = 60 nM T80276 CNL8D9 90664395 IC50 = 79 nM T80276 CMWN45 90664543 IC50 = 170 nM T80276 C47DQU 90664544 IC50 = 16 nM T80276 C0D1YZ 90664902 IC50 = 140 nM T80276 C08UWK 90665816 IC50 = 61000 nM T80276 CB1VI6 90665817 Ki = 0.57 nM T80276 CQ72ZV 90667915 IC50 = 1580 nM T80276 C38CHG 90667916 IC50 = 1400 nM T80276 CP0E4D 90667917 IC50 = 2890 nM T80276 CK69BQ 90667918 IC50 = 2490 nM T80276 CUG5O2 90667919 IC50 > 50000 nM T80276 CTS6E2 90667920 IC50 = 21630 nM T80276 CP1W6K 91755004 IC50 = 2.82 nM T80276 CMWB58 91757958 IC50 <= 10000 nM T80276 C3Y0DS 91801158 IC50 = 8.5 nM T80276 CAS7W6 91864650 IC50 = 150 nM T80276 C0Y8ZK 91933875 IC50 > 1000 nM T80276 C72IRG 118321317 IC50 = 6.87 nM T80276 C7EAJ0 118321318 IC50 = 23.3 nM T80276 CFQY64 118321319 IC50 = 145 nM T80276 C8AR0W 118321320 IC50 = 63.1 nM T80276 CBE08T 118321322 IC50 = 67 nM T80276 C67XRL 118321324 IC50 = 7.82 nM T80276 CH7MG0 118321327 IC50 = 8.41 nM T80276 C4CD6E 118321328 IC50 = 76.5 nM T80276 CXC7E3 118321354 IC50 = 82.4 nM T80276 C7KCB6 118321355 IC50 = 414 nM T80276 C67VQE 118341819 IC50 = 451 nM T80276 CC9P5H 118341835 IC50 = 201 nM T80276 CUMA23 118341844 IC50 = 115 nM T80276 C3IP9X 118341852 IC50 = 321 nM T80276 C6TI0Z 118341865 IC50 > 10000 nM T80276 C4U7NC 118341870 IC50 = 704 nM T80276 CVL03K 118341884 IC50 = 342 nM T80276 CPZN96 118341923 IC50 = 270 nM T80276 C9E3DU 118341927 IC50 = 475 nM T80276 C7EH3U 118352671 IC50 = 0.95 nM T80276 CM2DO8 118616331 IC50 = 54.1 nM T80276 CO0YC8 118616775 IC50 = 3.4 nM T80276 C42SYZ 118616923 IC50 = 98.8 nM T80276 CXA8N2 118616927 IC50 = 80.7 nM T80276 C84DGB 118616929 IC50 = 32.8 nM T80276 C8SRG9 118616951 IC50 = 67 nM T80276 CFQ71C 118616958 IC50 = 45 nM T80276 CU6E0P 118616985 IC50 = 141 nM T80276 C7WO2R 118617086 IC50 = 34.4 nM T80276 CVJU09 118617088 IC50 = 57.4 nM T80276 CQ7A1G 118617093 IC50 = 48.7 nM T80276 C6U0GQ 118617094 IC50 = 23.9 nM T80276 CB5XL3 118617097 IC50 = 48.8 nM T80276 CZ30BK 118617099 IC50 = 27.9 nM T80276 CGVH36 118617158 IC50 = 3.1 nM T80276 CCJ91U 118709071 IC50 = 12100 nM T80276 CL4U2W 118709072 IC50 = 1460 nM T80276 C2CE4Q 118709073 IC50 = 2880 nM T80276 C05EHL 118709074 IC50 = 330 nM T80276 CVS6W4 118709075 IC50 = 160 nM T80276 CZ5SO8 118709076 IC50 = 610 nM T80276 CRX24W 118709077 IC50 = 560 nM T80276 C9IUX6 118709078 IC50 = 2200 nM T80276 C7R9FA 118709079 IC50 = 6900 nM T80276 CY14MF 118709080 IC50 = 3800 nM T80276 CV2EJ7 118709081 IC50 = 2200 nM T80276 C9RF7I 118709082 IC50 = 4800 nM T80276 CVI98J 118709083 IC50 = 10100 nM T80276 CLEB72 118709084 IC50 = 1300 nM T80276 CV94YO 118709085 IC50 = 9400 nM T80276 CO3F4B 118709086 IC50 = 3400 nM T80276 CH4N9Y 118709087 IC50 = 8200 nM T80276 C8JZ7E 118709088 IC50 = 2500 nM T80276 C52YKH 118709089 IC50 = 4500 nM T80276 C94IZR 118709090 IC50 = 2400 nM T80276 C0UTL3 118709091 IC50 = 600 nM T80276 CH2ZF1 118709500 IC50 > 10000 nM T80276 C5BD7H 118709501 IC50 > 10000 nM T80276 C1W4CV 118709542 IC50 > 10000 nM T80276 C5SU1L 118709543 IC50 > 10000 nM T80276 CU0TC5 118709544 IC50 = 9700 nM T80276 CW5RO3 118709545 IC50 > 10000 nM T80276 C6EDP8 118709546 IC50 > 10000 nM T80276 C3MJ0O 118709547 IC50 > 10000 nM T80276 C6OX7W 118709548 IC50 > 10000 nM T80276 CANQ19 118709549 IC50 > 10000 nM T80276 C4Z3ME 118709550 IC50 > 10000 nM T80276 C0CLB5 118709551 IC50 > 10000 nM T80276 CTS23O 118709552 IC50 > 10000 nM T80276 CR6ML1 118709578 IC50 = 92 nM T80276 C0OH7I 118709579 IC50 = 1300 nM T80276 C73YIO 118709582 IC50 = 340 nM T80276 CGWX02 118709583 IC50 = 1200 nM T80276 C4AHL2 118711367 IC50 = 130 nM T80276 CR2V6S 118711765 IC50 = 5000 nM T80276 C9PWA0 118712008 IC50 > 1000 nM T80276 CVW2G8 118712009 IC50 > 1000 nM T80276 CTM26F 118712010 IC50 = 218 nM T80276 CH0K1V 118712011 IC50 = 38 nM T80276 CY5FS2 118712085 IC50 = 47.5 nM T80276 CPDT15 118712086 IC50 = 55.6 nM T80276 C2XC1O 118712087 IC50 = 117 nM T80276 CYCE79 118712088 IC50 = 632 nM T80276 CENO70 118712089 IC50 > 1000 nM T80276 CLC5I4 118715635 IC50 > 10000 nM T80276 CT6UF9 118715637 IC50 > 10000 nM T80276 CMG5I0 118715638 IC50 > 10000 nM T80276 CQX38N 118720611 IC50 = 40 nM T80276 CFP58Q 118720612 IC50 = 1100 nM T80276 CVIT16 118720879 IC50 > 10000 nM T80276 CJW06C 118720880 IC50 > 10000 nM T80276 C86RWG 118720882 IC50 > 10000 nM T80276 CYSD60 118720883 IC50 > 10000 nM T80276 CP6SR7 118721837 Ki = 16 nM T80276 CW4N7Q 118721838 Ki = 52 nM T80276 CZG78A 118721839 Ki = 56 nM T80276 C2BQS3 118721840 Ki = 7 nM T80276 C2T9RN 118721841 Ki = 72 nM T80276 C6GJ0Q 118721842 Ki = 105 nM T80276 C9RPN4 118721843 Ki = 113 nM T80276 CYNZ53 118721844 Ki = 67 nM T80276 C5R1VP 118721845 Ki > 4000 nM T80276 CB53EU 118728320 IC50 = 474 nM T80276 C6KJL1 118728321 IC50 = 283 nM T80276 CKJ3S6 118728322 IC50 = 181 nM T80276 CT0L3Y 118728325 IC50 = 127 nM T80276 CHS2E4 118728326 IC50 = 31 nM T80276 CRUP47 118728328 IC50 = 662 nM T80276 CQR41G 118728330 IC50 = 92 nM T80276 CN4Q9R 118728332 IC50 = 16 nM T80276 CDI10F 118728336 IC50 = 685 nM T80276 CHT6K9 118728811 Ki = 1800 nM T80276 CUA3Y2 118728812 Ki > 4000 nM T80276 CDQ78G 118728813 Ki = 850 nM T80276 CZ6XL7 118728814 Ki = 1500 nM T80276 CMO67K 118728815 Ki = 880 nM T80276 CR2M0Q 118728816 Ki > 4000 nM T80276 C62SCL 118728817 Ki = 1300 nM T80276 CSB30C 118728819 Ki > 4000 nM T80276 CV7XU8 118728820 Ki = 2600 nM T80276 C3J1EX 118728821 Ki > 4000 nM T80276 CIWB78 118728822 Ki > 4000 nM T80276 CP18SE 118728823 Ki > 4000 nM T80276 CM42CA 118728824 Ki > 4000 nM T80276 C9Q7CL 118728825 Ki > 4000 nM T80276 CCR3S0 118728826 Ki > 4000 nM T80276 CB1WC5 118729946 IC50 = 620 nM T80276 CQ4G9M 118729947 IC50 = 1600 nM T80276 C43IPJ 118729948 IC50 = 1370 nM T80276 C3I9CQ 118729949 IC50 = 1210 nM T80276 CZQ17M 118729950 IC50 = 830 nM T80276 CY60FC 118730033 IC50 = 118 nM T80276 CN3B4U 118730711 IC50 = 28 nM T80276 C0IL3N 118730712 IC50 = 110 nM T80276 C3CH1A 118730713 IC50 = 280 nM T80276 CHX5L9 118730714 IC50 = 18 nM T80276 CNJ32C 118730715 IC50 = 93 nM T80276 C1MKB3 118730716 IC50 = 10 nM T80276 C81RJA 118730717 IC50 = 970 nM T80276 CQCX41 118737057 IC50 > 10000 nM T80276 CFZ16R 118737301 IC50 <= 10000 nM T80276 C27CPQ 118737302 IC50 <= 10000 nM T80276 C59VXA 118737303 IC50 <= 10000 nM T80276 CGO1N4 118737304 IC50 <= 10000 nM T80276 CS85FM 118737305 IC50 <= 10000 nM T80276 C8UCO1 118737306 IC50 <= 10000 nM T80276 CR0BZ2 118737307 IC50 <= 10000 nM T80276 C3N4DJ 118737308 IC50 <= 10000 nM T80276 CGY5B1 118737309 IC50 <= 10000 nM T80276 CIN39H 121334370 Ki = 2 nM T80276 CJDS80 121334379 Ki = 633 nM T80276 CC1R8L 121334382 Ki = 15364 nM T80276 CU37QN 121334400 Ki = 2379 nM T80276 CSKB71 121334407 Ki = 8787 nM T80276 CM2ZS6 121334410 Ki > 20000 nM T80276 C4R7DN 121334420 Ki = 13.7 nM T80276 CK3G6P 121334425 Ki = 11.6 nM T80276 C01CNO 121334433 Ki = 11.1 nM T80276 CGCL96 121334436 Ki = 4.1 nM T80276 CB1L6S 121334438 Ki = 29 nM T80276 CV92TK 121334444 Ki = 18 nM T80276 CGD9K5 121334446 Ki = 25.8 nM T80276 CYTA71 121334474 Ki = 141 nM T80276 CH6Y9L 121334475 Ki = 1297 nM T80276 CHX60O 121334481 Ki = 2090 nM T80276 CYI09J 121334494 Ki = 32.2 nM T80276 CZ46TQ 121334504 Ki = 1.9 nM T80276 COZT28 121334509 Ki = 11.5 nM T80276 C1YQ8R 121334511 Ki = 632 nM T80276 C8M2ET 121334520 Ki = 4203 nM T80276 CBJ0C4 121406011 IC50 = 0.69 nM T80276 C91PVZ 121428416 IC50 = 15 nM T80276 CFN12W 121445751 IC50 = 2.3 nM T80276 C04NDW 121445810 IC50 = 8.2 nM T80276 C81IFQ 122163152 IC50 = 981 nM T80276 CL36RB 122178108 IC50 = 34.7 nM T80276 C4Q5KS 122178109 IC50 = 1.02 nM T80276 C2BV9G 122178110 IC50 = 0.095 nM T80276 CCHI06 122178111 IC50 = 51.7 nM T80276 C3FS4U 122178112 IC50 = 0.27 nM T80276 CT5J4A 122178113 IC50 = 0.07 nM T80276 C8NSE9 122178114 IC50 = 1228 nM T80276 C85GZQ 122178115 IC50 = 3494 nM T80276 C7X9HC 122178116 IC50 > 2500 nM T80276 C1MQ9F 122178117 IC50 = 43.1 nM T80276 C5PK7W 122178118 IC50 = 72.3 nM T80276 CN4R9Y 122178119 IC50 = 17 nM T80276 C2VGD5 122178120 IC50 = 2.07 nM T80276 CTE0F7 122178121 IC50 = 3.6 nM T80276 C3S2UI 122178122 IC50 = 1.3 nM T80276 C57MXE 122178123 IC50 = 1.7 nM T80276 C24XUZ 122178124 IC50 = 0.23 nM T80276 C3XMW0 122178125 IC50 = 0.3 nM T80276 C2P6KC 122178126 IC50 = 0.15 nM T80276 CN5AB3 122179486 IC50 = 13 nM T80276 CLEK13 122179487 IC50 = 9.6 nM T80276 CU1WJ9 122179488 IC50 = 13000 nM T80276 C2X1UO 122179489 IC50 = 46 nM T80276 C0OW8H 122179490 IC50 = 102 nM T80276 C0VD5F 122179491 IC50 = 12.6 nM T80276 CQ87FB 122179492 IC50 = 39.8 nM T80276 CBJ29X 122179493 IC50 = 2000 nM T80276 CA5N1B 122179494 IC50 = 16 nM T80276 CSTE64 122179689 IC50 = 1500 nM T80276 CE2FM7 122179690 IC50 = 1100 nM T80276 CZJ31R 122179691 IC50 = 790 nM T80276 CBOU30 122179692 IC50 = 1800 nM T80276 CKWC74 122179693 IC50 = 1100 nM T80276 C4CX7Z 122179694 IC50 = 6800 nM T80276 C48LYC 122179695 IC50 = 3100 nM T80276 C3D5QM 122179696 IC50 = 350 nM T80276 CW3DM7 122179697 IC50 = 6500 nM T80276 C6I3PB 122179698 IC50 > 10000 nM T80276 CCU6A4 122179699 IC50 = 1500 nM T80276 C7WMC3 122179700 IC50 = 1500 nM T80276 C86NOQ 122179701 IC50 = 2500 nM T80276 CAHY19 122179702 IC50 = 1600 nM T80276 C3O7CM 122179703 IC50 > 10000 nM T80276 CK2R4X 122179704 IC50 = 1700 nM T80276 CG96HD 122179705 IC50 = 4400 nM T80276 C1PK9L 122179706 IC50 > 1000 nM T80276 CEB69W 122179707 IC50 = 2900 nM T80276 CK97EL 122179708 IC50 = 3900 nM T80276 C0ZA4C 122179709 IC50 = 900 nM T80276 CU93YJ 122179710 IC50 > 10000 nM T80276 C0KTH8 122179711 IC50 = 490 nM T80276 CN9I1C 122179712 IC50 = 1800 nM T80276 C65OGI 122179713 IC50 = 850 nM T80276 C92AZK 122179714 IC50 = 1200 nM T80276 CWL43Z 122179715 IC50 = 4800 nM T80276 C50VNH 122179716 IC50 = 6500 nM T80276 COW37C 122179717 IC50 = 6400 nM T80276 CG5N9E 122179718 IC50 = 510 nM T80276 CB14FW 122179719 IC50 = 810 nM T80276 CHZ3S1 122179720 IC50 = 570 nM T80276 CEG8Y6 122179721 IC50 = 1360 nM T80276 CG5P3J 122179722 IC50 > 10000 nM T80276 CZH3T1 122179723 IC50 = 600 nM T80276 C10FGR 122179724 IC50 = 9000 nM T80276 CS85CU 122181413 IC50 = 16 nM T80276 CJ4T5W 122181414 IC50 = 27 nM T80276 CK8L4D 122181415 IC50 = 21 nM T80276 CQS67B 122181416 IC50 = 29 nM T80276 CB2AG9 122181417 IC50 = 280 nM T80276 CFET49 122181418 IC50 = 64 nM T80276 CQU14E 122181419 IC50 = 6 nM T80276 C58XRY 122184465 IC50 = 1584.89 nM T80276 C16ALM 122184466 IC50 = 1258.93 nM T80276 CIX19J 122184467 IC50 = 2511.89 nM T80276 CDZY02 122184468 IC50 = 63095.73 nM T80276 CTH70U 122184469 IC50 = 5011.87 nM T80276 C9ZXR7 122184470 IC50 = 1995.26 nM T80276 CNJ9Z4 122184471 IC50 = 6309.57 nM T80276 CMCP83 122184472 IC50 = 3162.28 nM T80276 CS41EG 122184473 IC50 = 1000 nM T80276 CZ36GL 122184474 IC50 = 1995.26 nM T80276 CU4ZT6 122184475 IC50 = 158489.32 nM T80276 C3H9PR 122184476 IC50 = 1258.93 nM T80276 CU40TW 122184477 IC50 = 2511.89 nM T80276 C8IK9C 122184478 IC50 = 1995.26 nM T80276 CAMD31 122184479 IC50 = 39810.72 nM T80276 C1F9RK 122184480 IC50 = 501.19 nM T80276 C7XW1K 122184481 IC50 = 10000 nM T80276 CRUX54 122184482 IC50 > 100000 nM T80276 CQ7W0P 122184526 IC50 = 1995.26 nM T80276 CA5YB2 122184529 IC50 = 6309.57 nM T80276 C64YPH 122184530 IC50 = 12589.25 nM T80276 C4AGX5 122184531 IC50 = 12589.25 nM T80276 CQL4K5 122184532 IC50 = 12589.25 nM T80276 CRKV74 122184533 IC50 = 15848.93 nM T80276 CX14YD 122184534 IC50 = 10000 nM T80276 CM6A4S 122184535 IC50 = 12589.25 nM T80276 CF86YS 122184536 IC50 = 7943.28 nM T80276 CH08SN 122184537 IC50 = 2511.89 nM T80276 CYRH97 122184538 IC50 = 6309.57 nM T80276 CD4W0Z 122184539 IC50 = 25118.86 nM T80276 CH8Y3Q 122184540 IC50 > 199526.23 nM T80276 CDA85R 122184541 IC50 > 199526.23 nM T80276 CF36XJ 122184542 IC50 > 199526.23 nM T80276 CQ6O7H 122184543 IC50 = 79432.82 nM T80276 CS4MN0 122184544 IC50 = 100000 nM T80276 CIB7W6 122184765 IC50 = 2820000 nM T80276 C4TVZ2 122184939 IC50 = 50 nM T80276 CVU7J2 122184940 IC50 = 90 nM T80276 C3TC0S 122184941 IC50 = 230 nM T80276 CQ20LR 122184942 IC50 = 1100 nM T80276 CWAG25 122184943 IC50 = 330 nM T80276 C74BUG 122184944 IC50 = 6000 nM T80276 C60RQI 122184945 IC50 = 80 nM T80276 CG3FO0 122184946 IC50 = 20 nM T80276 CMCL25 122184947 IC50 = 320 nM T80276 C72ZBC 122184948 IC50 = 110 nM T80276 CS5ED7 122184949 IC50 = 270 nM T80276 CXSL28 122184950 IC50 = 20 nM T80276 CWE3S6 122184951 IC50 = 10000 nM T80276 C25RKV 122184952 IC50 = 30 nM T80276 CPGO90 122184953 IC50 = 290 nM T80276 C93BNI 122185247 IC50 = 110 nM T80276 CW17SR 122185248 IC50 = 90 nM T80276 C8V9LF 122185249 IC50 = 4400 nM T80276 CZA26E 122185250 IC50 = 2200 nM T80276 CKT74G 122185265 IC50 = 7 nM T80276 CJ6C1O 122185267 IC50 = 14 nM T80276 CL0ZB6 122185870 IC50 = 980 nM T80276 CH2B5D 122185879 IC50 = 490 nM T80276 C9MIL3 122188249 IC50 = 271 nM T80276 C53AYQ 122188250 IC50 > 10000 nM T80276 CZO41H 122188251 IC50 > 10000 nM T80276 CLW25J 122188252 IC50 = 4350 nM T80276 C23PIE 122188253 IC50 > 10000 nM T80276 CE41KZ 122188254 IC50 > 10000 nM T80276 CHQT85 122188255 IC50 > 10000 nM T80276 CLAD59 122188256 IC50 > 10000 nM T80276 CI0W3V 122188257 IC50 = 4544 nM T80276 C3BXR2 122188258 IC50 = 5373 nM T80276 C67GYV 122188259 IC50 > 10000 nM T80276 CE81FB 122188260 IC50 = 7840 nM T80276 CG8VX5 122188261 IC50 > 10000 nM T80276 C9ZKA1 122188262 IC50 > 10000 nM T80276 CQF9I2 122188263 IC50 > 10000 nM T80276 COGF57 122188264 IC50 > 10000 nM T80276 CV8D3O 122188265 IC50 > 10000 nM T80276 CPQ89G 122188266 IC50 = 2960 nM T80276 CA4LH8 122188267 IC50 = 2963 nM T80276 CO9LT3 122188268 IC50 = 9430 nM T80276 CRH4E1 122188269 IC50 = 29 nM T80276 CXT3E9 122188270 IC50 = 81 nM T80276 CVEB28 122188271 IC50 = 902 nM T80276 C5E7WK 122188272 IC50 = 233 nM T80276 CWIR28 122188273 IC50 = 1240 nM T80276 CB6I5A 122188274 IC50 = 1030 nM T80276 CA8VH1 122188275 IC50 = 198 nM T80276 C1XAP9 122188276 IC50 = 327 nM T80276 C0BLT6 122188277 IC50 > 10000 nM T80276 CA6V5M 122188278 IC50 > 10000 nM T80276 CP9H3I 122188279 IC50 = 900 nM T80276 CV89ZC 122188280 IC50 = 1870 nM T80276 C2D5TF 122188281 IC50 > 10000 nM T80276 C93VST 122188282 IC50 = 194 nM T80276 C5FGI7 122188283 IC50 = 1070 nM T80276 CJY4C1 122188365 IC50 = 164 nM T80276 CJ82KW 122658866 IC50 = 680 nM T80276 C6YKO2 122658900 IC50 = 100 nM T80276 C1GH7B 122658923 IC50 > 20000 nM T80276 C2K9RM 122658945 IC50 = 200 nM T80276 CPTY78 124518210 IC50 = 820 nM T80276 C98DKI 127025346 IC50 = 5.5 nM T80276 CZDE86 127025619 IC50 > 100 nM T80276 CE2Q0R 127025620 IC50 = 37 nM T80276 CHM90W 127025621 IC50 = 70 nM T80276 CD7PN9 127025622 IC50 = 61 nM T80276 CBXJ67 127025628 IC50 = 2 nM T80276 C4Y7MN 127026222 IC50 = 32 nM T80276 CH7XY2 127026223 IC50 = 3.7 nM T80276 C5ZA0Q 127026224 IC50 = 33 nM T80276 CK9QU6 127026225 IC50 = 3.9 nM T80276 CB53ZX 127028515 IC50 = 690 nM T80276 CB9VY8 127028516 IC50 = 6720 nM T80276 C7IRF3 127029060 IC50 = 31 nM T80276 CS10AW 127029061 IC50 = 13 nM T80276 CDBS37 127029062 IC50 = 33 nM T80276 C64QWJ 127029063 IC50 = 11 nM T80276 CSV3R7 127029064 IC50 = 4.2 nM T80276 CV8AR2 127029085 Ki = 0.3 nM T80276 CP9B3A 127029332 IC50 > 10000 nM T80276 C4QKS1 127029333 IC50 > 10000 nM T80276 CBK8M2 127029338 IC50 = 74 nM T80276 CF78AE 127029339 IC50 > 10000 nM T80276 CAD38Y 127029440 IC50 = 4230 nM T80276 C6IDU4 127029598 IC50 = 1655 nM T80276 C1LW8M 127029599 IC50 = 142 nM T80276 CQ89TJ 127029600 IC50 = 778 nM T80276 CYP64N 127029601 IC50 = 2170 nM T80276 C7ZQE2 127029605 IC50 = 406 nM T80276 CY1CJ7 127029606 IC50 = 393 nM T80276 C1ZJW0 127029607 IC50 = 232 nM T80276 C3RP0D 127029608 IC50 = 609 nM T80276 C27ATB 127029609 IC50 = 419 nM T80276 CZ75CL 127029610 IC50 = 49 nM T80276 CR17GV 127029715 IC50 > 10000 nM T80276 CVBF01 127030212 IC50 = 650 nM T80276 C1ON3I 127030553 IC50 = 1180 nM T80276 CG35HU 127031182 IC50 = 270 nM T80276 CS12RU 127031435 IC50 = 2.2 nM T80276 CK7MR3 127032676 IC50 = 80 nM T80276 CGKR53 127032915 IC50 = 1500 nM T80276 C68TYB 127033266 IC50 = 1100 nM T80276 CV4BK1 127033886 IC50 = 1060 nM T80276 C41YQI 127035981 IC50 = 2427 nM T80276 C72NPR 127039226 IC50 = 3300 nM T80276 CL0ZU8 127040691 IC50 = 2800 nM T80276 CB0G7Z 127040692 IC50 > 10000 nM T80276 C3ZXT2 127040693 IC50 = 10000 nM T80276 CY6NM3 127040694 IC50 > 10000 nM T80276 C05MRE 127042767 IC50 = 3000 nM T80276 C4L9TC 127042949 IC50 = 10000 nM T80276 CG8DA9 127045861 IC50 = 300 nM T80276 CVF8Z9 127045862 IC50 = 3.5 nM T80276 CH68NT 127046076 IC50 = 44 nM T80276 CA2XD5 127046077 IC50 = 219 nM T80276 COJ68G 127046117 IC50 = 10 nM T80276 C34REM 127046317 IC50 = 16 nM T80276 CC4ND8 127046862 IC50 = 115 nM T80276 CO4N3J 127047042 IC50 = 54000 nM T80276 CY2P1X 127047138 IC50 = 10 nM T80276 CZ2R0C 127047140 IC50 = 6 nM T80276 CL18YE 127047185 IC50 = 38000 nM T80276 C8TIY1 127047186 IC50 = 37000 nM T80276 CVC5W1 127047187 IC50 = 19000 nM T80276 CW5X1G 127047188 IC50 = 44000 nM T80276 CT89GI 127047683 IC50 = 16 nM T80276 C7D0FN 127047685 IC50 = 5 nM T80276 CN94CQ 127047797 IC50 = 7 nM T80276 CJT02N 127048971 Ki = 5 nM T80276 CT98ID 127049341 Ki = 5 nM T80276 C9NO8C 127049342 Ki = 3 nM T80276 C1A0HV 127049343 Ki = 3 nM T80276 C18NHD 130302549 IC50 <= 10000 nM T80276 CL13RZ 130302558 IC50 <= 10000 nM T80276 CF5JZ3 130302563 IC50 <= 10000 nM T80276 CD46EL 130302605 IC50 <= 10000 nM T80276 CNI8M6 130302620 IC50 <= 10000 nM T80276 CI6WN9 130302651 IC50 <= 10000 nM T80276 C5ZP0L 130302658 IC50 <= 10000 nM T80276 CW61SG 130302663 IC50 <= 10000 nM T80276 CB27ZG 130302668 IC50 <= 10000 nM T80276 C5VYM6 130302674 IC50 <= 10000 nM T80276 C0FQR2 130302675 IC50 <= 10000 nM T80276 CB34HQ 130302676 IC50 <= 10000 nM T80276 CQR1I8 130302685 IC50 <= 10000 nM T80276 C17DZF 130302698 IC50 <= 10000 nM T80276 CBC6W7 130302701 IC50 <= 10000 nM T80276 CBT21G 130302702 IC50 <= 10000 nM T80276 CDZ45O 130302703 IC50 <= 10000 nM T80276 C2GWU8 130302709 IC50 <= 10000 nM T80276 CV3M6Y 130302710 IC50 <= 10000 nM T80276 C39UQN 130302731 IC50 <= 10000 nM T80276 CL9O8X 130302732 IC50 <= 10000 nM T80276 CL69GM 130302740 IC50 <= 10000 nM T80276 CH8YK9 130302741 IC50 <= 10000 nM T80276 CQR2W9 130302781 IC50 <= 10000 nM T80276 C9HC8A 130302803 IC50 <= 10000 nM T80276 CIK25W 130302809 IC50 <= 10000 nM T80276 CI08PF 130332501 IC50 <= 10000 nM T80276 C1H4UT 130332505 IC50 <= 10000 nM T80276 CZPI64 130332579 IC50 <= 10000 nM T80276 CDS9F3 130332582 IC50 <= 10000 nM T80276 C3G0HF 130332585 IC50 <= 10000 nM T80276 CX13UC 130332620 IC50 <= 10000 nM T80276 CED6F3 130332657 IC50 <= 10000 nM T80276 C47CAY 130421765 IC50 > 31622.78 nM T80276 C84YKI 130422161 IC50 > 31622.78 nM T80276 CK68CA 130453737 IC50 = 3800 nM T80276 CUO41K 130470684 IC50 = 445 nM T80276 CP32GB 132005220 IC50 = 730 nM T80276 CUN18W 132005225 IC50 = 55 nM T80276 CD84OI 132005228 IC50 = 53 nM T80276 C7ASP9 132005246 IC50 = 70 nM T80276 CBY49C 132156028 Ki = 20.8 nM T80276 C4M8WN 132209922 IC50 = 57 nM T80276 CFI23B 132210082 IC50 = 59 nM T80276 CH8DP7 132220479 IC50 = 370 nM T80276 C4Q5LF 132471857 IC50 = 10 nM T80276 CI6ZL8 132551695 IC50 >= 10000 nM T80276 CJE34F 132597748 IC50 = 14180 nM T80276 CCV46G 132606879 IC50 = 100 nM T80276 CV2PK1 134129977 IC50 = 111 nM T80276 CBR3Z9 134130128 IC50 = 67 nM T80276 C1LZP4 134131157 IC50 = 72 nM T80276 CFG90E 134132909 IC50 = 693 nM T80276 C4YNH0 134134126 IC50 = 218 nM T80276 C0EK8P 134134680 IC50 = 220 nM T80276 CLDS18 134135780 IC50 = 240 nM T80276 C0SE2M 134136023 IC50 = 2.5 nM T80276 C0A1UM 134138053 IC50 = 148 nM T80276 CQ2S4X 134138703 IC50 = 5080 nM T80276 CL3Q6G 134140420 IC50 = 888 nM T80276 CDJ10M 134142931 IC50 = 676 nM T80276 CUE85S 134143151 IC50 > 50000 nM T80276 CQ9G7H 134145670 IC50 = 127 nM T80276 C6G8EJ 134146051 IC50 = 47000 nM T80276 CIPL93 134147099 IC50 = 842 nM T80276 C8ITR3 134147904 IC50 = 43800 nM T80276 CG2T3L 134148055 IC50 = 1.1 nM T80276 CXA3V0 134148445 IC50 = 3230 nM T80276 CXU92M 134150578 IC50 = 491 nM T80276 CG8LE2 134151667 IC50 < 10000 nM T80276 CK43EY 134152988 IC50 = 424 nM T80276 CS2QP7 134154582 IC50 = 126 nM T80276 C2QGB3 134156160 IC50 = 1380 nM T80276 C42RJH 134157534 IC50 = 2611 nM T80276 CJXA12 134611894 IC50 > 31622.78 nM T80276 CX0UR7 134694318 IC50 = 2110 nM T80276 CBQ4J0 134956039 IC50 >= 25000 nM T80276 C9FUK2 135151360 IC50 = 14200 nM T80276 CJ1IZ5 135197550 IC50 = 3.3 nM T80276 C7Z9FJ 135197555 IC50 = 1.6 nM T80276 CI4SB8 135197556 IC50 = 4.8 nM T80276 C1TRQ4 135197560 IC50 = 1.2 nM T80276 CY1D0K 135197566 IC50 = 1.4 nM T80276 CT0GQ6 135197577 IC50 = 1.4 nM T80276 CQ3O1E 135197578 IC50 = 1.2 nM T80276 CMAP54 135197583 IC50 = 1.1 nM T80276 CB09NO 135197588 IC50 = 1.2 nM T80276 CQU0O6 135197590 IC50 = 1.5 nM T80276 CI65TH 135197591 IC50 = 4.1 nM T80276 CHCG03 135197593 IC50 = 0.95 nM T80276 C87VKA 135197594 IC50 = 0.96 nM T80276 C85UTD 135197595 IC50 = 1.8 nM T80276 CK7AW8 135197596 IC50 = 2.5 nM T80276 C6DY0Z 135197598 IC50 = 1.8 nM T80276 C05KVB 135197599 IC50 = 9.8 nM T80276 CA7R8Y 135197601 IC50 = 2 nM T80276 CP36TS 135197602 IC50 = 1.4 nM T80276 C0ZNA8 135197604 IC50 = 6.6 nM T80276 C06VRX 135197607 IC50 = 2.6 nM T80276 CDC5N3 135197609 IC50 = 1.1 nM T80276 CJTB73 135197628 IC50 = 1.4 nM T80276 C4RIL3 135197630 IC50 = 0.95 nM T80276 CKX2N5 135197633 IC50 = 0.83 nM T80276 CQXS07 135197635 IC50 = 1 nM T80276 CE2LG0 135197639 IC50 = 0.73 nM T80276 C7KXF1 135197643 IC50 = 0.8 nM T80276 C60NDC 135197644 IC50 = 1.7 nM T80276 CY1FC7 135197646 IC50 = 1.1 nM T80276 CFKB59 135197651 IC50 = 1.4 nM T80276 C1CR6U 135197655 IC50 = 1.1 nM T80276 CV27KJ 135197680 IC50 = 1.6 nM T80276 C5W8NU 135197682 IC50 = 1 nM T80276 CW6O9Z 135197693 IC50 = 0.7 nM T80276 C96FJI 135197694 IC50 = 11 nM T80276 CK4MW9 135197700 IC50 = 5.4 nM T80276 CY38TL 135391000 IC50 = 766.6 nM T80276 COG86Z 135397763 IC50 = 2511.89 nM T80276 CWL67T 135397764 IC50 = 630.96 nM T80276 CX8AI4 135398491 IC50 = 11 nM T80276 C6AZ2R 135435018 IC50 > 25118.86 nM T80276 CPW45Y 135452024 IC50 = 23000 nM T80276 C3QJ8W 135566371 IC50 = 9000 nM T80276 CEK31P 135566415 IC50 > 20000 nM T80276 C24ZGX 135566644 IC50 = 10000 nM T80276 C2QDV5 135566741 IC50 = 2138 nM T80276 C0TE5S 135651612 IC50 = 300 nM T80276 C2UN0D 135742360 IC50 = 14200 nM T80276 CU29YK 135750268 IC50 = 510 nM T80276 CD6UJ5 135857414 IC50 = 3565 nM T80276 C41HNJ 135857415 IC50 = 720 nM T80276 C8K3HJ 135911704 IC50 > 10000 nM T80276 C02PHA 135927892 IC50 = 25118.86 nM T80276 CS8T3D 135927897 IC50 > 25118.86 nM T80276 C12UDA 135947972 IC50 = 92 nM T80276 CN42ZS 135947973 IC50 = 480 nM T80276 CF8AO3 135947974 IC50 = 296 nM T80276 CW08GJ 135947976 IC50 = 80 nM T80276 C8O9HG 135947977 IC50 = 100000 nM T80276 CJN7E2 135947978 IC50 = 260 nM T80276 CFKH34 135947979 IC50 = 1300 nM T80276 C9OAV5 135986100 IC50 = 100000 nM T80276 C3USL8 135986101 IC50 > 100000 nM T80276 CG9PJ7 135993841 IC50 = 2150 nM T80276 C42STV 136013318 IC50 = 910 nM T80276 CT1K2H 136013322 IC50 = 6500 nM T80276 CP1US5 136041737 IC50 = 626 nM T80276 CXH63V 136041747 IC50 > 10000 nM T80276 C6B5TC 136041748 IC50 > 10000 nM T80276 CU6XG1 136041749 IC50 = 5460 nM T80276 C0U5DB 136041750 IC50 > 10000 nM T80276 C48KAQ 136041752 IC50 > 10000 nM T80276 C74PRL 136041753 IC50 > 10000 nM T80276 CT4FJ1 136041757 IC50 = 460 nM T80276 CCS2G6 136041761 IC50 = 9768 nM T80276 CEZP21 136041762 IC50 > 10000 nM T80276 CJ58TD 136041764 IC50 > 10000 nM T80276 CX67QW 136041765 IC50 = 6790 nM T80276 CK0H2Q 136041766 IC50 = 5725 nM T80276 CQP7B6 136041767 IC50 = 4353 nM T80276 CM65BS 136041773 IC50 = 1000 nM T80276 C6P7JB 136041775 IC50 = 5650 nM T80276 C5CJF7 136041776 IC50 > 10000 nM T80276 C3XIZ8 136041777 IC50 > 10000 nM T80276 C32LKO 136041785 IC50 = 9880 nM T80276 C90ARP 136041787 IC50 > 10000 nM T80276 CZ3BN1 136041792 IC50 = 2450 nM T80276 CG19DI 136041799 IC50 = 8400 nM T80276 CXJA29 136041804 IC50 = 2265 nM T80276 CHT31V 136041805 IC50 = 426 nM T80276 CO8C4J 136041817 IC50 = 569 nM T80276 C4QU6G 136041827 IC50 = 2020 nM T80276 CNE10X 136041834 IC50 = 2425 nM T80276 CS3AE1 136041847 IC50 = 2870 nM T80276 CZC47Y 136041848 IC50 = 2553 nM T80276 CM81HG 136044188 IC50 > 10000 nM T80276 CT6N1O 136044189 IC50 = 6900 nM T80276 C9PTA8 136044190 IC50 > 10000 nM T80276 CM1EN4 136044191 IC50 > 10000 nM T80276 C89CTO 136066004 IC50 = 6270 nM T80276 CLA3C2 136068720 IC50 = 15 nM T80276 CA91JG 136069599 IC50 = 217 nM T80276 CGAB91 136069600 IC50 = 1000 nM T80276 C3ZAW2 136069605 IC50 = 390 nM T80276 C8JXL5 136069609 IC50 = 1000 nM T80276 C9I0EQ 136069610 IC50 = 2375 nM T80276 C25EYJ 136069611 IC50 = 361 nM T80276 C2S5QF 136069615 IC50 = 660 nM T80276 CG1R7B 136087060 IC50 = 27 nM T80276 C48DBY 136118009 IC50 = 400 nM T80276 CHE5I7 136118010 IC50 = 26 nM T80276 CC4UM3 136176116 IC50 = 5503 nM T80276 CJRK81 136176117 IC50 = 314 nM T80276 C63IOS 136176118 IC50 = 4575 nM T80276 C3KW7H 136176119 IC50 > 10000 nM T80276 C69AKQ 136176120 IC50 = 7798 nM T80276 CF17KO 136176121 IC50 > 10000 nM T80276 CU3TE0 136176122 IC50 > 10000 nM T80276 C6C5KB 136176123 IC50 > 10000 nM T80276 C3X5KE 136176124 IC50 = 7150 nM T80276 CA8C5E 136176125 IC50 > 10000 nM T80276 C5OMG2 136176126 IC50 = 7754 nM T80276 CP2YM7 136176127 IC50 > 10000 nM T80276 C8XIJ0 136176128 IC50 = 4357 nM T80276 CUY8N4 136176129 IC50 = 3333 nM T80276 C3J4ME 136176130 IC50 > 10000 nM T80276 CR1NZ2 136176131 IC50 > 10000 nM T80276 C4WG2F 136176132 IC50 > 10000 nM T80276 CJ8EC5 136176139 IC50 > 10000 nM T80276 CQ84IZ 136180335 Ki > 4000 nM T80276 C04XFY 136180790 IC50 > 10000 nM T80276 C1LK9U 136183381 IC50 = 85 nM T80276 C27TKQ 136196449 IC50 = 960 nM T80276 CC1X7G 136227360 IC50 = 12200 nM T80276 C5KW4P 136227361 IC50 = 283000 nM T80276 CK9S4X 136229137 IC50 = 4300 nM T80276 CAI9M5 136229138 IC50 = 3000 nM T80276 C8M5HN 136229139 IC50 = 7900 nM T80276 C5ZFP8 136229140 IC50 = 4880 nM T80276 CS1X6P 136229141 IC50 = 4520 nM T80276 CXQG23 136229142 IC50 = 3380 nM T80276 C07INE 136229143 IC50 = 2200 nM T80276 CHXY59 136229144 IC50 = 82600 nM T80276 CVHL13 136229146 IC50 = 160000 nM T80276 CDEX74 136229147 IC50 = 840 nM T80276 CRJ47T 136229148 IC50 = 62300 nM T80276 C7S1YJ 136230225 IC50 > 10000 nM T80276 C3Q6ED 136230226 IC50 = 6218 nM T80276 CKPF02 136230227 IC50 > 10000 nM T80276 CZY9O0 136230228 IC50 = 2273 nM T80276 CRET01 136230229 IC50 = 2373 nM T80276 CX1KI8 136230230 IC50 = 1905 nM T80276 C3Z5MH 136230231 IC50 = 3845 nM T80276 CUE6N8 136230232 IC50 = 831 nM T80276 C8Q1AP 136230233 IC50 = 1900 nM T80276 C70RXE 136230234 IC50 = 3460 nM T80276 C4W0KN 136230235 IC50 = 4140 nM T80276 CMZN01 136230236 IC50 = 8143 nM T80276 CCU0H5 136241428 IC50 = 138 nM T80276 CF3DK1 136245085 IC50 = 18600 nM T80276 CEU87Z 136245089 IC50 = 10000 nM T80276 CI6HG4 136249373 IC50 = 45 nM T80276 CL4MO3 136249382 IC50 = 5421 nM T80276 C0GZV9 136254283 IC50 > 10000 nM T80276 CMWA86 136264282 IC50 = 322 nM T80276 CSD78N 136264452 IC50 = 1540 nM T80276 C1HI5T 136264454 IC50 = 86 nM T80276 CV3UE9 137333450 IC50 = 62.6 nM T80276 CH39TP 137453801 Ki = 6.8 nM T80276 C1EK8U 137453918 Ki = 4 nM T80276 CP34TI 137631388 IC50 = 610 nM T80276 CB5SZ7 137631459 IC50 >= 25000 nM T80276 CIX4S7 137633081 IC50 = 1584.89 nM T80276 C9GXM1 137635017 IC50 = 1995.26 nM T80276 C06BDR 137635072 IC50 = 180 nM T80276 C0L9UJ 137635168 IC50 >= 25000 nM T80276 CO8X7R 137636042 IC50 = 8 nM T80276 CMN6T7 137636115 IC50 = 624 nM T80276 CPJ43Y 137636841 IC50 = 1200 nM T80276 C8GQD5 137636872 IC50 = 6226 nM T80276 CC12YG 137638766 IC50 >= 50 nM T80276 CMZV19 137639099 IC50 = 31.62 nM T80276 CJ3LX4 137639119 IC50 = 1100 nM T80276 CS78JW 137639139 IC50 = 6 nM T80276 C4TSZ8 137639858 IC50 = 158.49 nM T80276 CA0QO6 137640453 IC50 = 591 nM T80276 CI0FJ1 137641054 IC50 < 1000 nM T80276 CQ8X0E 137641383 IC50 = 8300 nM T80276 C0I6RQ 137641405 IC50 = 316.23 nM T80276 C5X3TH 137642662 IC50 = 3300 nM T80276 C8M9TX 137642801 IC50 = 630 nM T80276 CP4DI5 137643070 IC50 > 10000 nM T80276 CP3JK1 137643598 IC50 = 316.23 nM T80276 CF74MH 137643612 IC50 < 5000 nM T80276 CI9D4L 137645884 IC50 > 10000 nM T80276 CFB71W 137646194 IC50 < 5000 nM T80276 CY20QZ 137646387 IC50 >= 15000 nM T80276 C5ERV3 137646413 IC50 = 930 nM T80276 CZC27Y 137646667 IC50 = 63.1 nM T80276 C3TXN9 137647591 IC50 = 3110 nM T80276 CPX42N 137647765 IC50 = 270 nM T80276 C9FTP7 137648413 IC50 = 22000 nM T80276 C4Z0NQ 137648826 IC50 = 3162.28 nM T80276 CS4AP5 137649695 IC50 >= 5000 nM T80276 CSML14 137649696 IC50 = 1486 nM T80276 C37WLI 137650083 IC50 < 10 nM T80276 CHT1R8 137650579 IC50 = 316.23 nM T80276 C2O7XP 137651832 IC50 >= 25000 nM T80276 CN78RE 137653565 IC50 = 100 nM T80276 CD19ZS 137654937 IC50 = 250 nM T80276 C4N5LS 137655123 IC50 = 158.49 nM T80276 CV3TF0 137655436 IC50 >= 50 nM T80276 CRK30E 137655634 IC50 >= 25000 nM T80276 CHV26G 137655828 IC50 = 54 nM T80276 CTB78E 137655854 IC50 = 5 nM T80276 CJB90Y 137656872 IC50 = 20 nM T80276 CE9H8D 137657006 IC50 = 1995.26 nM T80276 C41OPW 137658031 IC50 = 3981.07 nM T80276 CA5C1Q 137658327 IC50 >= 5000 nM T80276 C6BF8E 137658458 IC50 = 1700 nM T80276 C13NKV 137658788 IC50 >= 25000 nM T80276 C03JHP 137659077 IC50 >= 15000 nM T80276 CP5K4E 137660883 IC50 = 1481 nM T80276 C1OLQ3 137660961 IC50 = 1584.89 nM T80276 CM6FS2 137661095 IC50 = 501.19 nM T80276 C8R3JK 137661301 IC50 = 63.1 nM T80276 CBXL91 137661615 IC50 < 25000 nM T80276 CA3C4O 138454792 IC50 = 42 nM T80276 CKDZ26 138504497 IC50 = 2200 nM T80276 C1NQ0F 139207772 Ki = 990 nM T80276 C3O5IA 139207773 Ki = 920 nM T80276 CKLH15 139207774 Ki = 150 nM T80276 C26NWP 139486659 Ki = 64 nM T80276 C7ZAQ1 141406387 IC50 = 40780 nM T80276 C7NUI8 141406388 IC50 = 44660 nM T80276 CQYI18 141406390 IC50 = 3690 nM T80276 CUA1D0 141406392 IC50 = 52870 nM T80276 CP0R6Y 141406393 IC50 = 730 nM T80276 C1EVQ0 141406394 IC50 = 9680 nM T80276 C2QP0F 141406396 IC50 = 6480 nM T80276 CY2M0B 141406399 IC50 = 1440 nM T80276 CC3OU2 141406400 IC50 = 27670 nM T80276 CKV13Y 141406404 IC50 = 12540 nM T80276 C3Q1VL 141419885 IC50 = 25.6 nM T80276 C3EJX8 141419888 IC50 = 26.7 nM T80276 CKX4P3 141446054 IC50 > 158489.32 nM T80276 CV54CS 141471198 IC50 = 1.1 nM T80276 C25HYI 141471200 IC50 = 1.3 nM T80276 CBXR10 141471201 IC50 = 2.2 nM T80276 CW2IP3 141471202 IC50 = 9.3 nM T80276 CG8IF9 141471203 IC50 = 2.3 nM T80276 C27RTX 141471204 IC50 = 2.2 nM T80276 C7FB1M 141471208 IC50 = 1.6 nM T80276 C32ZOH 141471209 IC50 = 3 nM T80276 C8P1QH 141481226 IC50 = 1250 nM T80276 CZS03J 141509623 IC50 = 254 nM T80276 CQ34YR 142506035 IC50 = 387 nM T80276 CU03GW 142506036 IC50 = 75 nM T80276 C74MXW 142506065 IC50 = 52 nM T80276 CX6BQ7 142506102 IC50 = 13 nM T80276 CC6MD0 142506155 IC50 = 186 nM T80276 C05QOM 142506157 IC50 = 517 nM T80276 CT3U9R 142506192 IC50 = 9 nM T80276 C1T3IQ 142506210 IC50 = 122 nM T80276 CEGV67 142506220 IC50 = 266 nM T80276 CP5HF8 142506225 IC50 = 422 nM T80276 C1U3CA 142506238 IC50 = 50 nM T80276 C8FZE6 142608579 Ki = 780 nM T80276 C7QMG9 145108300 IC50 = 2.3 nM T80276 C2YN6G 145949270 IC50 = 24 nM T80276 C3TCJ7 145949910 IC50 = 2847 nM T80276 C1X2TN 145950166 IC50 = 125 nM T80276 CT6AR4 145950273 IC50 = 38 nM T80276 CI40JE 145951013 IC50 = 59.8 nM T80276 C6YT8E 145951131 IC50 = 6660 nM T80276 CFW62M 145951569 IC50 = 62.1 nM T80276 CTGX37 145951752 IC50 = 31 nM T80276 CHA84K 145951830 IC50 > 10000 nM T80276 CT4I9A 145952160 IC50 = 29.5 nM T80276 C91GVH 145952598 IC50 = 24.7 nM T80276 C1W0GJ 145952796 IC50 = 25118.86 nM T80276 CIK0D1 145952943 IC50 = 86 nM T80276 CVMF13 145953272 IC50 = 1448 nM T80276 CYL5T1 145953372 IC50 <= 10000 nM T80276 CP14AV 145953653 IC50 = 28 nM T80276 CY8D5Q 145953886 IC50 = 27.7 nM T80276 C3ZUW8 145954195 IC50 = 78.2 nM T80276 C1NJB7 145955070 IC50 = 7.5 nM T80276 CRHE01 145955133 IC50 <= 10000 nM T80276 C7MP9Z 145955279 IC50 = 41.2 nM T80276 C7K8VT 145955565 IC50 = 105.8 nM T80276 CPU4X2 145955670 IC50 = 129.1 nM T80276 C3ST5Y 145955693 IC50 = 19.9 nM T80276 C1VH5X 145955836 IC50 = 52.8 nM T80276 CBP1S9 145955956 IC50 = 16 nM T80276 C7K2YF 145956631 IC50 <= 10000 nM T80276 CQW74M 145956683 IC50 = 14.8 nM T80276 CJ1F6A 145956725 IC50 = 328.5 nM T80276 CHO1M9 145956818 IC50 = 18 nM T80276 C12IFO 145956886 IC50 = 33.9 nM T80276 CS4O8H 145957011 IC50 = 90 nM T80276 C9O2PL 145958063 IC50 = 22.8 nM T80276 CQH01X 145958257 IC50 <= 10000 nM T80276 C3DGU7 145958571 IC50 < 10 nM T80276 C9NS6T 145958690 IC50 = 43 nM T80276 C7ZO9V 145959196 IC50 = 1017 nM T80276 CSC81H 145959429 IC50 = 15.6 nM T80276 C0S1YM 145959980 IC50 = 222 nM T80276 CT3I2R 145960112 IC50 = 75.9 nM T80276 C8MJ9X 145960272 IC50 = 73.2 nM T80276 CF36RA 145961004 IC50 = 53.5 nM T80276 CHF56O 145961403 IC50 = 2020 nM T80276 C2GT9Y 145961404 IC50 = 6940 nM T80276 CAI0D6 145963117 IC50 = 17.7 nM T80276 CQTC03 145967732 IC50 = 5.6 nM T80276 C46INV 145967893 IC50 = 1.3 nM T80276 CVI41O 145968143 IC50 = 7 nM T80276 CN20TV 145968302 IC50 = 1.6 nM T80276 C1P7GV 145968320 IC50 = 2.8 nM T80276 C8AK3I 145968593 IC50 = 6.1 nM T80276 C45OUF 145969270 IC50 = 4.5 nM T80276 C3W9NF 145969494 IC50 = 1.5 nM T80276 C97IKW 145969580 IC50 = 25.4 nM T80276 CK82QG 145969816 IC50 = 165 nM T80276 C71YAK 145970017 IC50 = 290000 nM T80276 CMR92A 145970234 IC50 = 2.2 nM T80276 CDI8N7 145970354 IC50 = 2.4 nM T80276 C40ATS 145970821 IC50 = 1 nM T80276 CZ98FH 145971490 IC50 = 1224 nM T80276 CTB97Z 145971948 IC50 = 66 nM T80276 CGQJ04 145972017 IC50 = 604.5 nM T80276 CZ9G6E 145974533 IC50 = 48.3 nM T80276 C3LR4O 145976442 IC50 = 317 nM T80276 CZ1T9X 145979969 Ki = 68.6 nM T80276 CZ8E2C 145980061 EC50 > 500000 nM T80276 C03BJC 145980560 Ki = 23.7 nM T80276 CGA83C 145981271 IC50 > 30000 nM T80276 CVR1X3 145981509 Ki = 2230 nM T80276 C8DCW3 145981748 EC50 = 15100 nM T80276 CJ1G9L 145981832 Ki = 693 nM T80276 CPZS56 145982349 EC50 = 550 nM T80276 CH90CT 145983168 IC50 = 26.7 nM T80276 CH6X1R 145983184 Ki > 20000 nM T80276 CJU02I 145983624 IC50 = 11814 nM T80276 CVS2U0 145983808 IC50 = 31291 nM T80276 C05LJH 145984149 EC50 = 1200 nM T80276 CF8MR5 145986347 IC50 = 250000 nM T80276 CKU3Q0 145986508 EC50 = 6300 nM T80276 CD70WO 145986565 Ki = 5668 nM T80276 C5R6BS 145987142 IC50 = 300 nM T80276 C6D8QS 145987359 Ki = 129 nM T80276 C7KVT0 145987381 IC50 = 240 nM T80276 C4BWJ3 145987648 Ki > 20000 nM T80276 C9TYO4 145988008 Ki = 81.3 nM T80276 C58ALF 145988716 EC50 = 2100 nM T80276 C12GWM 145988761 EC50 = 58400 nM T80276 CW7IF0 145989521 EC50 = 9700 nM T80276 CD6GZ1 145989663 EC50 > 500000 nM T80276 C8GPL7 145989970 EC50 = 7100 nM T80276 CAZ8S0 145990081 EC50 = 5100 nM T80276 C8FZY6 145990358 EC50 = 39300 nM T80276 CV47FK 145990785 EC50 = 42700 nM T80276 C32MJQ 145990827 Ki > 20000 nM T80276 CH6P5O 145991719 EC50 = 8900 nM T80276 CSYC93 145991982 Ki = 2190 nM T80276 C6OI8X 145992071 EC50 > 500000 nM T80276 C2J0XO 145992074 IC50 = 9000 nM T80276 CA0J2B 145992083 Ki = 4632 nM T80276 C2BJW1 145992739 EC50 = 6370 nM T80276 C36RTB 145993509 IC50 = 78.2 nM T80276 C6XC9B 145993646 EC50 > 500000 nM T80276 CI6GL9 145993781 EC50 = 900 nM T80276 C8WK1V 145993856 EC50 = 242300 nM T80276 C8X2IT 145996536 IC50 = 2200 nM T80276 C6RPG0 146014481 IC50 = 5.623 nM T80276 C59KOM 146585662 IC50 = 47 nM T80276 CFQO97 146585699 IC50 = 444 nM T80276 C0GMR1 146585718 IC50 = 392 nM T80276 CI85VS 146731761 IC50 = 9 nM T80276 C4MC0S 149169124 IC50 = 450 nM T80276 CVW62P 149242889 IC50 = 8120 nM T80276 CN87RZ 149370890 IC50 = 300 nM T80276 CK4FJ1 149556361 IC50 = 3840 nM T80276 C8UQL4 153940691 IC50 = 950 nM T80276 CMZ68Q 153940692 IC50 = 42 nM T80276 C5X7JK 154734328 IC50 = 3981.07 nM T80276 C69VNW 155510695 IC50 = 15848.93 nM T80276 C6ISA2 155510865 IC50 = 5.1 nM T80276 CDT8F2 155510913 IC50 = 501.19 nM T80276 C1ZXV2 155511261 IC50 = 0.69 nM T80276 C1OR2T 155511706 IC50 = 1000 nM T80276 CGH08E 155511904 IC50 = 2290.87 nM T80276 C8VDK1 155511906 IC50 = 2.3 nM T80276 CG07YP 155512189 IC50 = 707.95 nM T80276 CZJ9D6 155512258 IC50 = 2861 nM T80276 C7FO1Y 155512340 IC50 = 54 nM T80276 CG9I4X 155512515 IC50 = 120 nM T80276 CR1Z8A 155512529 IC50 = 633 nM T80276 C8UYW4 155512651 IC50 = 630.96 nM T80276 CQZY50 155512775 IC50 = 39.81 nM T80276 C5V2GO 155512947 IC50 = 6309.57 nM T80276 C1DIT4 155513047 IC50 = 100 nM T80276 C8PG6Z 155513084 IC50 = 2511.89 nM T80276 CK63OT 155513410 IC50 = 4.786 nM T80276 CMZR80 155513562 IC50 = 331.13 nM T80276 C45SYX 155513615 IC50 = 4.5 nM T80276 C4UZI2 155514046 IC50 = 25118.86 nM T80276 C17NTI 155514706 Ki > 10000 nM T80276 CBH57O 155514764 IC50 = 3981.07 nM T80276 CXVL19 155514838 IC50 = 116 nM T80276 C5C9EG 155515047 IC50 = 630.96 nM T80276 CEFS61 155515135 IC50 = 1550 nM T80276 CX72DF 155515279 IC50 = 5011.87 nM T80276 CR1XO3 155515353 IC50 = 25118.86 nM T80276 CBK3C9 155515384 Ki = 3200 nM T80276 C0AXF7 155515394 IC50 = 630.96 nM T80276 CXTC52 155515425 IC50 = 25118.86 nM T80276 CTJ43N 155515666 IC50 = 7.1 nM T80276 C7Q3FR 155515734 IC50 = 2511.89 nM T80276 CFD72J 155516184 IC50 = 143 nM T80276 CL45GQ 155516260 IC50 = 1584.89 nM T80276 C30ZFN 155516445 IC50 = 501.19 nM T80276 CJDG04 155516604 IC50 = 63.1 nM T80276 CNP25D 155516982 IC50 = 1.8 nM T80276 CYO19V 155517071 IC50 = 125.89 nM T80276 CYWX76 155517213 IC50 = 501.19 nM T80276 C0D3NR 155517424 IC50 = 25118.86 nM T80276 C7SEB5 155517457 IC50 = 0.6 nM T80276 C4G8YN 155517534 IC50 = 358 nM T80276 C8FWK7 155517588 IC50 = 50.12 nM T80276 CV0EF2 155518789 IC50 = 1202.26 nM T80276 CW7OM6 155518918 IC50 = 190 nM T80276 C8XCP4 155519431 IC50 = 162 nM T80276 CC51GM 155519635 IC50 = 125.89 nM T80276 C81SOG 155520064 IC50 = 213 nM T80276 CQEK39 155520373 IC50 = 0.5 nM T80276 C5D6YX 155521099 IC50 = 650 nM T80276 CEA3M1 155521494 IC50 = 31.62 nM T80276 CBSR95 155522042 IC50 = 1170 nM T80276 CZO7Q8 155522149 IC50 = 114 nM T80276 CABC57 155522182 Ki > 10000 nM T80276 C9FNJ8 155523062 IC50 = 43 nM T80276 CCGW06 155523124 IC50 = 3162.28 nM T80276 CZ3FC8 155523374 Ki = 19.9 nM T80276 C4TLQ7 155523447 IC50 > 10000 nM T80276 C37RVF 155523599 IC50 = 399 nM T80276 C4H2AB 155524238 IC50 = 19.95 nM T80276 CP18VT 155524467 IC50 = 10000 nM T80276 CF40DG 155524748 IC50 = 7.7 nM T80276 CUP7L2 155524901 IC50 = 251.19 nM T80276 CYK1M8 155524976 IC50 = 2.3 nM T80276 CJMD34 155525139 Ki > 10000 nM T80276 C2BL5I 155525312 IC50 = 39.81 nM T80276 CE2OM4 155525333 IC50 = 7943.28 nM T80276 C10RZQ 155525477 IC50 = 1258.93 nM T80276 CF76OV 155525717 IC50 = 1.8 nM T80276 C0UA4D 155525996 IC50 = 50.12 nM T80276 C31XHG 155526170 IC50 = 94 nM T80276 CNHS85 155526193 IC50 = 15848.93 nM T80276 C3EAR8 155526323 IC50 = 501.19 nM T80276 CC9W3J 155527176 IC50 = 4 nM T80276 C9PI3H 155527271 IC50 = 43 nM T80276 C82NUW 155527501 IC50 = 83 nM T80276 CK07GS 155527559 IC50 = 183 nM T80276 CX12MK 155527651 IC50 = 42 nM T80276 CF2P3Q 155527936 Ki > 20000 nM T80276 C3JFZ8 155528005 IC50 = 12 nM T80276 CE64FQ 155528066 IC50 = 106 nM T80276 C08KBN 155528302 IC50 = 0.9 nM T80276 CPLV31 155528423 IC50 = 91.2 nM T80276 C5Z7SQ 155528446 IC50 = 346.74 nM T80276 C8Z3TK 155528581 IC50 = 794.33 nM T80276 C0B2NV 155528644 IC50 = 12700 nM T80276 C9OVL5 155528904 Ki = 85 nM T80276 C9L6OC 155529247 IC50 = 226 nM T80276 C2FE1S 155529479 IC50 = 31.62 nM T80276 C70MEU 155529500 IC50 = 72 nM T80276 CM6E3Q 155529607 IC50 = 2.8 nM T80276 CB90AR 155529643 IC50 = 1584.89 nM T80276 CFV1S0 155529706 IC50 = 123 nM T80276 C14QOF 155530163 IC50 = 1584.89 nM T80276 C4I5UP 155530224 IC50 = 63.1 nM T80276 CTQ2P0 155530465 IC50 = 43 nM T80276 CX6N3Y 155531155 IC50 = 31.62 nM T80276 C9AXO7 155531257 IC50 = 251.19 nM T80276 C7U8YQ 155531296 IC50 = 0.9 nM T80276 CE7Q6O 155531509 IC50 = 30 nM T80276 CDI4V8 155531526 IC50 = 32 nM T80276 CH8ST1 155531582 IC50 = 323.59 nM T80276 CE6QP1 155532037 IC50 = 501.19 nM T80276 CIM18N 155532540 IC50 = 7500 nM T80276 C3XFB8 155532820 IC50 = 10 nM T80276 C0GR1J 155533050 IC50 = 119.5 nM T80276 CQS8P1 155533070 IC50 = 398.11 nM T80276 C0SZR9 155533335 IC50 = 7943.28 nM T80276 CAT9V1 155533370 IC50 = 829 nM T80276 C67ERP 155533384 IC50 = 125.89 nM T80276 CL8OM7 155533564 IC50 = 1767 nM T80276 CBM24U 155533579 IC50 = 3162.28 nM T80276 CR5H8B 155533591 IC50 = 3162.28 nM T80276 CA7T0Y 155533911 IC50 = 6180 nM T80276 CN1ST4 155534269 IC50 = 1995.26 nM T80276 CBEG39 155534594 IC50 = 316.23 nM T80276 CQ2N7Y 155534617 IC50 = 7 nM T80276 CCGS79 155535013 IC50 = 68 nM T80276 CS0L4T 155535224 IC50 = 1 nM T80276 C6O8JB 155535273 IC50 = 1.1 nM T80276 CN6KJ5 155535520 IC50 = 1584.89 nM T80276 C8N6MT 155535532 IC50 = 15848.93 nM T80276 C5F2TY 155535537 IC50 = 3162.28 nM T80276 CKB2U4 155535691 IC50 = 25.12 nM T80276 CY7X3M 155535740 IC50 = 19.95 nM T80276 C70UDF 155536179 IC50 = 794.33 nM T80276 CEJ6L1 155536226 IC50 = 18.2 nM T80276 CNB24M 155536473 IC50 = 1584.89 nM T80276 C2CG1A 155537016 IC50 = 6309.57 nM T80276 CX9EO1 155537184 IC50 = 41 nM T80276 C5A2WC 155537194 IC50 = 73 nM T80276 C1Y9MS 155537503 Ki > 10000 nM T80276 CS24EV 155537776 IC50 = 4900 nM T80276 C8AJ6C 155538256 IC50 = 21.8 nM T80276 CQ1E6H 155538266 IC50 = 19.95 nM T80276 CZ19AN 155538609 IC50 = 98 nM T80276 CV7HK0 155538979 IC50 = 2.6 nM T80276 CHR8M1 155538990 IC50 = 8910 nM T80276 CC1BG2 155539321 IC50 > 10000 nM T80276 CF20PS 155539394 IC50 = 1584.89 nM T80276 C7TB4V 155539520 IC50 = 0.4 nM T80276 C8LKW4 155540264 IC50 = 1584.89 nM T80276 CE8TV9 155541005 Ki > 10000 nM T80276 CI8XL2 155541479 IC50 = 1400 nM T80276 C2D4ZP 155541609 IC50 > 31622.78 nM T80276 C57MVO 155542051 IC50 = 12589.25 nM T80276 C5OQ3G 155542658 IC50 = 82 nM T80276 CYB90C 155542790 Ki > 10000 nM T80276 C8OC2P 155542800 IC50 = 90 nM T80276 CVNR95 155542898 IC50 = 84 nM T80276 CV5L6B 155543139 Ki = 250 nM T80276 C1SY0G 155543154 IC50 = 29200 nM T80276 CJE20U 155543234 IC50 = 691.83 nM T80276 C1JRK8 155543277 IC50 > 31622.78 nM T80276 C1UNH0 155543517 IC50 = 3162.28 nM T80276 CY48WX 155543524 IC50 > 10000 nM T80276 CZY0N4 155543588 IC50 = 18 nM T80276 CJB8C9 155543659 IC50 = 40 nM T80276 C5MYJ2 155543736 IC50 = 10000 nM T80276 CSUW45 155544033 IC50 = 34 nM T80276 CV2G1W 155544267 IC50 = 0.66 nM T80276 C1NF0S 155544279 IC50 = 8380 nM T80276 CX1C8I 155544561 IC50 = 4600 nM T80276 CBN29V 155544583 IC50 = 36 nM T80276 COGF23 155544916 IC50 > 31622.78 nM T80276 C98FXC 155544955 IC50 = 2371 nM T80276 C5IVX6 155544961 Ki = 37 nM T80276 CW3K4F 155545182 IC50 = 3162.28 nM T80276 C4TYN3 155545535 IC50 > 31622.78 nM T80276 CE02BC 155545624 IC50 = 2511.89 nM T80276 CTSW53 155546042 IC50 = 9800 nM T80276 CS0I4N 155546205 IC50 = 44.67 nM T80276 CQ6J7U 155546361 IC50 = 20 nM T80276 C8SQA2 155546999 IC50 = 7.943 nM T80276 CJ1E0T 155547067 Ki = 15.2 nM T80276 CKR36G 155547524 Ki = 31.4 nM T80276 CIQ8G6 155547573 IC50 = 3.9 nM T80276 CI6KO7 155548518 IC50 = 199.53 nM T80276 C6JCV4 155548973 Ki = 2600 nM T80276 CL4F8P 155549003 IC50 = 15.85 nM T80276 CJWV35 155549094 Ki = 2200 nM T80276 CFM6A5 155549676 IC50 = 3008 nM T80276 C4PEJ5 155549895 IC50 = 8300 nM T80276 CGNF42 155549917 Ki = 4643 nM T80276 CFP94J 155550309 IC50 = 316.23 nM T80276 CQ5OD0 155550395 IC50 = 8 nM T80276 CCX5E2 155550788 IC50 = 2600 nM T80276 C0JEH6 155551208 IC50 = 169.82 nM T80276 C5HR2W 155551907 IC50 > 31622.78 nM T80276 CK1JR7 155551961 IC50 = 0.7 nM T80276 CF8D9H 155552080 Ki = 31 nM T80276 CJ75BO 155552100 IC50 = 452 nM T80276 CL04BD 155554125 IC50 = 465 nM T80276 CX9C6O 155554180 IC50 = 199.53 nM T80276 CC13QL 155555170 IC50 = 908 nM T80276 C2OGW1 155555483 IC50 = 67 nM T80276 C84KXJ 155555515 IC50 = 131.83 nM T80276 C3UP9A 155555623 IC50 = 6309.57 nM T80276 C1TW9S 155555707 IC50 = 30.2 nM T80276 C62XMN 155555936 IC50 = 5.3 nM T80276 CRO5Z3 155556073 IC50 = 2047 nM T80276 CH2P4T 155556124 IC50 > 50118.72 nM T80276 C3BK7O 155556309 Ki = 684 nM T80276 CNW48Z 155556396 IC50 = 2.1 nM T80276 CIU29Z 155556576 IC50 = 5800 nM T80276 CM3LI6 155556593 IC50 = 3896 nM T80276 CZ8CX1 155556887 IC50 = 251.19 nM T80276 CG2FS6 155557123 IC50 = 3981.07 nM T80276 CFS63H 155557182 IC50 = 5760 nM T80276 C0FE4G 155557988 IC50 = 855 nM T80276 CR8J0E 155558167 IC50 = 39.81 nM T80276 C52TSP 155558262 IC50 = 191 nM T80276 CB4A1O 155558535 IC50 = 2511.89 nM T80276 CZMI26 155558737 IC50 = 25118.86 nM T80276 CX70UY 155558767 IC50 = 102 nM T80276 CS70ER 155559192 IC50 = 183 nM T80276 CMKY39 155559468 IC50 = 19952.62 nM T80276 CGH85A 155560338 IC50 = 48 nM T80276 CVG49I 155560688 IC50 = 2630 nM T80276 C5S7AL 155560766 IC50 = 79.43 nM T80276 C2OT6K 155560767 IC50 = 6309.57 nM T80276 CLO3B1 155561152 IC50 = 259 nM T80276 C8XS0L 155561165 IC50 = 125.89 nM T80276 C72CQG 155561233 IC50 = 125.89 nM T80276 C1INL7 155561328 IC50 = 199.53 nM T80276 CQ0T4D 155561330 IC50 = 73 nM T80276 C98FHW 155561366 IC50 = 7300 nM T80276 C1QZ8A 155561726 IC50 = 0.63 nM T80276 CUGI82 155561991 IC50 = 6100 nM T80276 C4GXV3 155562151 Ki > 10000 nM T80276 CB1T2W 155562315 IC50 > 31622.78 nM T80276 CX6U2T 155562388 IC50 = 3981.07 nM T80276 CN4B3D 155562639 IC50 = 7943.28 nM T80276 C0JRI5 155562814 IC50 = 562.34 nM T80276 C6RV0H 155563416 Ki = 4600 nM T80276 CCF4W2 155563986 IC50 = 3981.07 nM T80276 CC04GI 155564488 IC50 = 19.95 nM T80276 CHK4E8 155565269 IC50 = 251.19 nM T80276 C7PXA0 155565551 IC50 = 794.33 nM T80276 CY4N7O 155565715 IC50 > 31622.78 nM T80276 CVQ6Z4 155565763 IC50 = 398.11 nM T80276 CKJ36M 155565775 IC50 = 51 nM T80276 CMK4I3 155565845 IC50 = 3162.28 nM T80276 C59VPW 155565958 IC50 = 3162.28 nM T80276 CAP9F2 155566187 IC50 = 42 nM T80276 CM7E2G 155566279 IC50 = 3981.07 nM T80276 C1BUC4 155566417 IC50 = 3175 nM T80276 C9HR5K 155566863 IC50 = 19952.62 nM T80276 C6V3EC 155567228 IC50 = 195 nM T80276 C3XMB6 155567232 Ki = 1000 nM T80276 C6DQ2X 155567318 IC50 = 1.3 nM T80276 C9KQW3 155567372 IC50 = 410 nM T80276 C1HQ5J 155568324 IC50 = 8591 nM T80276 CLA46O 155568356 IC50 = 100 nM T80276 C7SLR8 155568452 IC50 = 794.33 nM T80276 CT15RN 155568479 IC50 = 6309.57 nM T80276 C1S8ZB 155568922 IC50 = 247 nM T80276 CTG81X 155569017 Ki = 731 nM T80276 C14LVO 155569074 IC50 = 79.43 nM T80276 C6NY3Z 155569079 IC50 = 43.65 nM T80276 CFWP17 155569113 IC50 = 4941 nM T80276 CXBZ67 155569362 IC50 > 31622.78 nM T80276 CUH38L 155569363 IC50 > 10000 nM T80276 C4H0NE 155569598 IC50 = 316.23 nM T80276 CQ6C3M 155569679 IC50 = 58 nM T80276 COIQ01 44577787 IC50 > 10000 nM T80276 CR9C5Y 44577828 IC50 = 262 nM T80276 CHB1K5 44577829 IC50 = 174 nM T80276 D00GQM 25069592 IC50 = 2894 nM T80276 D00HSJ 10275789 IC50 = 0.5 nM T80276 D00JIV 51033720 Ki = 0.6 nM T80276 D00ZIK 9908783 IC50 > 200000 nM T80276 D02TSN 46244454 IC50 = 13000 nM T80276 D03EHM 24905142 IC50 = 52 nM T80276 D03QQH 16760391 IC50 = 32000 nM T80276 D05BPX 9901372 IC50 = 2 nM T80276 D05USL 5278396 IC50 = 458 nM T80276 D06DNH 9907093 IC50 = 1000 nM T80276 D06HVH 54613583 IC50 > 9100 nM T80276 D06PWI 42623951 IC50 > 10000 nM T80276 D07JKB 135955185 IC50 = 667 nM T80276 D07PMP 44187953 IC50 = 1 nM T80276 D07QJJ 289 IC50 = 33000 nM T80276 D08KSQ 11637090 IC50 > 10000 nM T80276 D08NQM 5289247 IC50 = 60 nM T80276 D09FBN 135955186 IC50 = 2538 nM T80276 D0AH8Q 25074311 IC50 = 640 nM T80276 D0F1SI 25074312 IC50 = 2381 nM T80276 D0H0HR 49836027 EC50 = 1800 nM T80276 D0H2CM 135565635 IC50 = 2000 nM T80276 D0N2LW 11324758 IC50 > 100000 nM T80276 D0P5TI 58441401 EC50 = 10 nM T80276 D0Q5FJ 11185819 IC50 > 100000 nM T80276 D0R0TW 11964036 IC50 = 4 nM T80276 D0R2UG 52936849 IC50 = 0.8 nM T80276 D0S5YV 6852167 IC50 = 39 nM T80276 D0T0BY 10039361 IC50 > 100000 nM T80276 D0TC5H 16049458 IC50 = 150 nM T80276 D0W1ST 9860529 IC50 = 13000 nM T80276 D0W8XH 9884685 IC50 = 2 nM T80276 D0X7TB 10017389 IC50 = 2400 nM T80276 D0Y1DR 46225260 IC50 = 2330 nM T80276 D0Y3OO 11327430 IC50 = 130 nM T80276 D0Z5KQ 8400 IC50 = 2120000 nM T56143 D00HGB 4488 EC50 = 1110 nM T56143 D02TJS 54676038 Ki = 39 nM T56143 D04AIT 5280445 EC50 = 3200 nM T56143 D0B9GH 2882 EC50 = 52 nM T56143 D0G5UB 2161 EC50 = 4000 nM T56143 D0G7IY 27503 EC50 = 1260 nM T56143 D0J1VY 5281081 EC50 = 5660 nM T56143 D0K8KX 5280343 EC50 = 5930 nM T56143 D0OG3K 44564 EC50 = 4000 nM T56143 D0PQ3G 3440 Ki = 3270 nM T56143 D0Y7PG 4659569 EC50 = 7440 nM T56143 D00YPW 135399235 EC50 = 110 nM T56143 D08LVF 5464105 EC50 = 820 nM T56143 CTS0K5 1493 EC50 = 31100 nM T56143 CI9TK0 3884 EC50 = 2840 nM T56143 C7OG9U 6191 EC50 = 58500 nM T56143 C8BQT7 9492 EC50 = 52600 nM T56143 CZ2C1F 10800 EC50 = 6910 nM T56143 CT65JS 11312 EC50 = 18200 nM T56143 CG4DE1 11348 EC50 = 112000 nM T56143 CRJ4V2 11872 EC50 = 5270 nM T56143 CVR65K 13681 EC50 = 5450 nM T56143 C6S5PV 40119 EC50 = 3400 nM T56143 CXJV17 73157 EC50 = 2390 nM T56143 CAWR46 92934 Ki = 9860 nM T56143 CB1VR4 119405 EC50 = 23200 nM T56143 CIM16P 271643 EC50 = 13520 nM T56143 C20QIO 633803 EC50 = 2350 nM T56143 CH7NC6 657910 EC50 = 2020 nM T56143 CUXA91 660319 EC50 = 42400 nM T56143 CD48TY 694463 EC50 = 10760 nM T56143 CB5DI3 725495 EC50 = 1749.85 nM T56143 C7F0BP 782693 EC50 = 21430 nM T56143 C7A3EH 1230851 EC50 > 40000 nM T56143 CA1Y2P 1230852 EC50 > 40000 nM T56143 C46QDC 1231538 EC50 = 550 nM T56143 C8KD9F 1281702 EC50 > 10000 nM T56143 C7L1HF 1920221 EC50 > 40000 nM T56143 C4G9CE 1941471 EC50 > 40000 nM T56143 C3P9EW 1951822 EC50 > 40000 nM T56143 C6NLQ0 2286812 Ki = 8.76 nM T56143 CRK06N 2295463 Ki = 50.8 nM T56143 CR7AO8 3254949 EC50 = 6 nM T56143 CYI94Z 3495594 EC50 = 8660 nM T56143 C20LJC 4679731 EC50 > 40000 nM T56143 CY2KU8 4921319 EC50 = 190 nM T56143 C2BWF7 5066064 IC50 = 8610 nM T56143 CSU5J3 5098885 EC50 = 54 nM T56143 C94SUH 5328791 EC50 = 9800 nM T56143 C1MKI4 5346366 IC50 = 7230 nM T56143 CH4R8E 5491415 EC50 = 390 nM T56143 C93EYT 9581011 Ki = 42.2 nM T56143 CRYT62 9990345 IC50 = 12100 nM T56143 CQR16D 10339735 EC50 > 40000 nM T56143 CTZ5K7 10857978 EC50 = 1390 nM T56143 C9W7JL 10868388 EC50 = 44060 nM T56143 CT8G0R 11338511 IC50 > 10000 nM T56143 CD5RP7 11674067 IC50 = 1940 nM T56143 C3L6FB 11748721 IC50 > 10000 nM T56143 CH1B9N 12138434 EC50 = 15300 nM T56143 CKJ0I9 12138435 EC50 = 32 nM T56143 CBF0U1 12403015 EC50 = 13 nM T56143 C52FWD 13950957 IC50 = 3760 nM T56143 CXZJ39 13950958 EC50 = 149.97 nM T56143 C7Q8HG 14950683 IC50 > 10000 nM T56143 CHS4M8 15774807 EC50 = 45400 nM T56143 CVB93E 15774808 EC50 = 43500 nM T56143 CQ4L2F 16103462 EC50 = 61 nM T56143 CCL16V 16103465 EC50 = 6000 nM T56143 CTA4I1 16103482 EC50 = 3440 nM T56143 CKT1A8 20259231 EC50 = 7350 nM T56143 C5P0QE 20486870 EC50 = 6760 nM T56143 C7E1ZI 21236027 IC50 = 3750 nM T56143 CYE24K 21337669 EC50 = 45900 nM T56143 CZL70J 21337670 EC50 = 6600 nM T56143 COS8P6 21337671 IC50 = 48900 nM T56143 C08OIG 21982642 Ki = 13600 nM T56143 CFP9S1 44157038 EC50 > 40000 nM T56143 CUG4T6 45093111 EC50 = 16200 nM T56143 C1Q5TM 45489602 EC50 = 645.65 nM T56143 CX9M3E 49837912 EC50 > 40000 nM T56143 CVQM43 51035368 EC50 > 40000 nM T56143 C65GEF 51035373 EC50 > 40000 nM T56143 C9YIZ5 52914819 EC50 > 40000 nM T56143 C6S9YI 52914822 EC50 > 40000 nM T56143 C3Y4DQ 52914826 EC50 > 40000 nM T56143 CC4U3O 53245521 EC50 > 40000 nM T56143 C3WTY4 53245542 EC50 > 40000 nM T56143 CE7A9B 53245571 EC50 > 40000 nM T56143 CH4EO6 53245574 EC50 > 40000 nM T56143 CMJ62D 53245590 EC50 > 40000 nM T56143 CQHV82 53245615 EC50 > 40000 nM T56143 C69HCK 53245626 EC50 > 40000 nM T56143 CE5Y0F 53257379 EC50 = 11100 nM T56143 C4DA0K 53258793 EC50 = 1460 nM T56143 CP7E4Z 53258795 EC50 = 1890 nM T56143 CK41VO 53258796 EC50 = 2310 nM T56143 CRWP87 53258898 EC50 = 4560 nM T56143 C5UQ7A 53258899 EC50 = 9400 nM T56143 C0HI5E 54758538 EC50 > 40000 nM T56143 CZ63WS 54758539 EC50 > 40000 nM T56143 CC6F4U 56593272 EC50 > 40000 nM T56143 CY5VX7 56593273 EC50 > 40000 nM T56143 C1RJX8 56593274 EC50 > 40000 nM T56143 CX1N3I 56593278 EC50 > 40000 nM T56143 CMF4H8 56593279 EC50 > 40000 nM T56143 CB75SU 56593281 EC50 > 40000 nM T56143 C2J7VC 56593282 EC50 > 40000 nM T56143 CA9OV0 56593283 EC50 > 40000 nM T56143 C2FHP7 56593284 EC50 > 40000 nM T56143 CNG48L 56593288 EC50 > 40000 nM T56143 CY1N5C 56593289 EC50 > 40000 nM T56143 C7ZL2B 56593290 EC50 > 40000 nM T56143 CD06NY 56593291 EC50 > 40000 nM T56143 CQ60KY 56593292 EC50 > 40000 nM T56143 CNB83L 56593293 EC50 > 40000 nM T56143 CQ6HS2 56646802 EC50 = 3350 nM T56143 CGJ03F 57134579 EC50 = 29990 nM T56143 C9Y6QT 66561717 EC50 = 16 nM T56143 CO3GD2 66561718 EC50 = 240 nM T56143 CA4E6U 66561793 EC50 = 630 nM T56143 C6KCE4 70681838 EC50 = 1290 nM T56143 CU59AR 70681839 EC50 = 8370 nM T56143 C8YPM0 70682865 EC50 = 4100 nM T56143 C2L0KC 70682869 EC50 = 10300 nM T56143 CU6YA0 70683937 EC50 = 510 nM T56143 C0J5FL 70683938 EC50 = 9780 nM T56143 C6FA1D 70683939 EC50 = 950 nM T56143 CH2BJ9 70684936 EC50 = 6170 nM T56143 CD17GC 70686064 EC50 = 700 nM T56143 C16ZQW 70686065 EC50 = 370 nM T56143 CWP89L 70687102 EC50 = 10800 nM T56143 C4QS0U 70687103 EC50 = 1060 nM T56143 CEKR51 70687104 EC50 = 4360 nM T56143 C6Y0OK 70689180 EC50 = 43700 nM T56143 CTK9F7 70689183 EC50 = 84000 nM T56143 CN79MR 70689184 EC50 = 24900 nM T56143 CT7A8U 70689185 EC50 = 12900 nM T56143 C9PH0L 70690212 EC50 = 2630 nM T56143 CVNL36 70690213 EC50 = 5300 nM T56143 CZ80DG 70691265 EC50 = 39700 nM T56143 C7AY4F 70691267 EC50 = 2540 nM T56143 C1XJ0E 70691268 EC50 = 160 nM T56143 C1XCF9 70692386 EC50 = 260 nM T56143 C47MHF 70692387 EC50 = 11800 nM T56143 C0T2MV 70693381 EC50 = 20200 nM T56143 C0I7RX 70694439 EC50 = 1480 nM T56143 CY2IZ3 70695483 EC50 = 2480 nM T56143 C5IAX6 70696510 EC50 = 1030 nM T56143 C3NBP7 70697498 EC50 = 45700 nM T56143 CPJ6C2 70697499 EC50 = 17300 nM T56143 CN6TW5 71733647 Ki = 233 nM T56143 CN59OP 71733648 Ki = 119 nM T56143 CT6P5H 71733649 Ki = 4.12 nM T56143 C0V9LA 71733650 Ki = 11.5 nM T56143 CDO29X 71733651 Ki = 25.4 nM T56143 CDA14J 71733652 Ki = 138 nM T56143 CW79JG 71733653 Ki = 250 nM T56143 CQ28CY 71733743 Ki = 183 nM T56143 CA0S4Q 71733744 Ki = 5.5 nM T56143 CXQ8F9 71733745 Ki = 81.6 nM T56143 CQ30PL 71733746 Ki = 128 nM T56143 C2MV1Z 71733747 Ki = 4.79 nM T56143 CC9T2D 71733748 Ki = 0.938 nM T56143 C0X2OW 71733749 Ki = 2.18 nM T56143 C0TY2C 71733842 Ki = 148 nM T56143 C31ANM 71733843 Ki = 5.18 nM T56143 CO5R8A 71733844 Ki = 98.4 nM T56143 C2PZ4T 71733845 Ki = 331 nM T56143 CLKR10 71733846 Ki = 228 nM T56143 CI4A7M 71733847 Ki = 15 nM T56143 CU32CA 71733848 Ki = 1.12 nM T56143 CYEV04 71733937 Ki = 3710 nM T56143 CZ8IS9 71733938 Ki = 8060 nM T56143 CM7GX1 71733939 Ki = 56.8 nM T56143 CG8JP7 71733940 Ki = 25.7 nM T56143 CZL28N 71734939 Ki = 3010 nM T56143 CT3XR4 71734940 EC50 = 112 nM T56143 CQ6JB4 71734941 Ki = 18500 nM T56143 CF0EH5 71734942 Ki = 6770 nM T56143 C9VR1W 71734943 Ki = 18600 nM T56143 CKZO87 71734944 Ki = 3580 nM T56143 CIQ0X7 71734945 Ki = 2720 nM T56143 CRMI92 71734946 Ki = 714 nM T56143 CEAU94 71735030 Ki = 691 nM T56143 CQW63U 71735031 Ki = 3290 nM T56143 CA7C4D 71735032 Ki = 4780 nM T56143 C0YF7O 71735033 Ki = 4390 nM T56143 CGH9O0 71735034 Ki = 697 nM T56143 CUVE95 71735035 Ki = 10300 nM T56143 C0E5WK 71735036 Ki = 221 nM T56143 CFWZ35 73294319 Ki = 1.92 nM T56143 CG4T0Q 73294320 Ki = 1.37 nM T56143 CUDJ98 73294321 Ki = 1.64 nM T56143 CJ96BG 73294508 Ki = 0.589 nM T56143 CM3B6W 73294509 EC50 = 37.7 nM T56143 C1VFU0 73294510 Ki = 20.5 nM T56143 CG62IS 73346308 EC50 > 40000 nM T56143 CO8S0I 73347807 EC50 > 40000 nM T56143 CH2YN5 73349346 EC50 > 40000 nM T56143 C6V7YB 73350917 EC50 > 40000 nM T56143 C8PZ4T 73352405 EC50 > 40000 nM T56143 C4G6FB 73353870 EC50 > 40000 nM T56143 C5IVA1 73355398 EC50 > 40000 nM T56143 CGTQ84 73356947 EC50 > 40000 nM T56143 CQ91AR 73356948 EC50 > 40000 nM T56143 CQE10H 85468767 IC50 > 10000 nM T56143 CA0Y8G 85469571 EC50 > 10000 nM T56143 C31ZMH 90667661 EC50 > 10000 nM T56143 C0B6SI 110720191 EC50 = 17580 nM T56143 CA58HT 125756071 IC50 > 30000 nM T56143 CM1B0O 125759247 IC50 > 30000 nM T56143 C8CB5W 135403802 EC50 = 4700 nM T56143 CSL8M6 135468531 EC50 = 3.2 nM T56143 CWN95O 137632781 EC50 = 930 nM T56143 CJ0S2L 137632988 EC50 = 576.77 nM T56143 C2U6CI 137635873 IC50 = 13000 nM T56143 CQXA79 137636652 EC50 = 14760 nM T56143 CXA24V 137638263 IC50 > 30000 nM T56143 C7MOQ5 137641148 EC50 = 710 nM T56143 C8E6LD 137643028 IC50 > 30000 nM T56143 CEU1A3 137643561 EC50 = 9270 nM T56143 CB1YU4 137646097 EC50 = 2660 nM T56143 CPT5U1 137646246 EC50 = 51 nM T56143 CME8R4 137646699 IC50 = 5240 nM T56143 CCW49L 137647638 IC50 = 17000 nM T56143 CLOF69 137647862 EC50 = 2910 nM T56143 C8OI2S 137648473 EC50 = 330 nM T56143 C32HAK 137652009 IC50 = 13 nM T56143 CF2MV9 137653726 IC50 = 23 nM T56143 C3WE0F 137654727 IC50 = 590 nM T56143 C1LSM3 137655259 EC50 = 17700 nM T56143 CC0W5J 137657450 EC50 = 1409.29 nM T56143 CK0ZR2 137658268 EC50 = 2330 nM T56143 C1R2KJ 137658472 EC50 = 887.16 nM T56143 CS0TQ6 137658805 IC50 > 30000 nM T56143 C31GQK 137660898 IC50 > 30000 nM T56143 CY5OF6 137662152 EC50 = 5.781 nM T56143 CWL0Y7 145949189 EC50 = 199.53 nM T56143 C04WVZ 145950576 EC50 = 1060 nM T56143 CP28LU 145951357 EC50 = 310 nM T56143 CSW8N0 145951566 IC50 = 60 nM T56143 CYZ10U 145952039 IC50 = 400 nM T56143 C0FZ1V 145952453 EC50 = 870 nM T56143 C6W4KI 145952561 EC50 = 4600 nM T56143 CE6C5U 145952912 EC50 = 610 nM T56143 CJZ7A4 145953203 EC50 = 830 nM T56143 C3P8ND 145953959 EC50 = 3650 nM T56143 CQ1EG9 145954149 EC50 = 446.68 nM T56143 CD15GC 145954727 EC50 = 616.6 nM T56143 C4VGK3 145955027 IC50 = 260 nM T56143 CS41EH 145955278 EC50 = 2180 nM T56143 CH74KI 145956623 EC50 = 41 nM T56143 CWH7N2 145957901 IC50 = 110 nM T56143 CZGL43 145958445 EC50 = 2050 nM T56143 C0AY9R 145958495 EC50 = 436.52 nM T56143 CLT48F 145958540 EC50 = 520 nM T56143 CSYC98 145959306 EC50 = 1940 nM T56143 C1XPO0 145959592 IC50 = 510 nM T56143 CK54IU 145959908 EC50 = 870 nM T56143 CEK5F7 145971240 EC50 = 380 nM T56143 CTB5K0 145971442 EC50 = 58.88 nM T56143 CH5YN0 145971743 EC50 = 346.74 nM T56143 CPQ30F 145974046 IC50 = 360 nM T56143 D00YEV 5281605 EC50 = 10300 nM T56143 D01SHB 3845 EC50 = 39200 nM T56143 D04BYU 8546 EC50 = 2 nM T56143 D09AYR 3870203 EC50 = 22000 nM T56143 D0A1CM 5281855 EC50 = 110 nM T56143 D0H3NS 10752 EC50 = 92260 nM T56143 D0NJ4H 5281670 EC50 = 1330 nM T56143 D0T3PW 5281672 IC50 = 2120 nM T29741 D04AIT 5280445 IC50 = 850 nM T29741 D0K8KX 5280343 IC50 = 680 nM T29741 C0W4UD 3896 IC50 = 1340 nM T29741 C4SED3 1226613 IC50 > 100000 nM T29741 CBV4I8 1494838 Ki > 30000 nM T29741 C43XAE 1496853 Ki = 1845 nM T29741 CEB82A 1510303 Ki = 5232 nM T29741 C1DCS4 2538148 Ki = 880 nM T29741 CAUC54 3563087 Ki = 4729 nM T29741 CQ21NS 4112136 Ki = 373 nM T29741 CDG9Q7 4979726 Ki = 1208 nM T29741 C6JK3V 4979889 Ki = 5440 nM T29741 CH0JF4 5280417 IC50 = 1020 nM T29741 CO3A9X 5281604 IC50 = 740 nM T29741 C84ANP 5306234 Ki = 878 nM T29741 C6M9VU 5328657 IC50 = 1580 nM T29741 C1R9UM 6339420 Ki = 35600 nM T29741 CO4Z2V 7342677 Ki = 9490 nM T29741 C10SZX 10106602 IC50 = 960 nM T29741 CG1AS6 10333483 IC50 = 1270 nM T29741 CQ43JU 10426229 IC50 = 630 nM T29741 CWA2B6 12304323 IC50 = 830 nM T29741 CBK4Y5 16460081 Ki > 30000 nM T29741 CQ7EZ4 16460204 Ki = 4222 nM T29741 CO3NX2 16460217 Ki > 30000 nM T29741 CTFX75 16472615 Ki > 30000 nM T29741 CW4DN9 17609478 Ki = 3120 nM T29741 CUP1J6 21255453 IC50 = 1580 nM T29741 C4IDJ5 25014586 Ki = 173 nM T29741 CIYH60 45110789 Ki = 409 nM T29741 C1WEY5 46102359 Ki = 13100 nM T29741 C5CS1D 46182725 Ki = 285 nM T29741 C3KTQ1 46182771 Ki = 463 nM T29741 CB0OG9 46937440 IC50 = 260 nM T29741 CL53AP 46937441 IC50 = 590 nM T29741 CB0I5U 46937442 IC50 = 240 nM T29741 C6WRG9 49836177 Ki = 313 nM T29741 C9V3TW 49836178 Ki = 445 nM T29741 CM2T5K 49836179 Ki = 334 nM T29741 C1A9SY 49836180 Ki = 326 nM T29741 C6O8HA 49836181 Ki = 218 nM T29741 C6WXF8 49836182 Ki = 342 nM T29741 COU14A 49836183 Ki = 259 nM T29741 C0QF8E 49836288 Ki = 235 nM T29741 C9A5EB 49836289 Ki = 458 nM T29741 CA04IH 49836290 Ki = 165 nM T29741 CPOL41 49836291 Ki = 153 nM T29741 C3TX0L 49836292 Ki = 114 nM T29741 CDO7I4 49836293 Ki = 151 nM T29741 CY6Q7N 49836403 Ki = 65 nM T29741 C4Z1SQ 49836404 Ki = 172 nM T29741 CT2P4E 49836406 Ki = 95 nM T29741 CUSZ36 49836407 Ki = 82 nM T29741 CFI75Q 49836408 Ki = 114 nM T29741 C7QS9M 49836516 Ki = 128 nM T29741 C78BJV 49837377 Ki > 30000 nM T29741 CA3X5W 49837479 Ki > 30000 nM T29741 C8KN4E 49837572 Ki = 215 nM T29741 C97IML 49837573 Ki = 308 nM T29741 C6LHU2 49837574 Ki = 1947 nM T29741 CH29VP 49837575 Ki = 1418 nM T29741 C8TYU0 49837576 Ki = 2175 nM T29741 CX80UB 49837577 Ki = 213 nM T29741 CBI2W0 49837578 Ki = 3060 nM T29741 C7Z3BX 49837681 Ki = 293 nM T29741 C4YQ0N 49837682 Ki = 340 nM T29741 C1U8BK 49837683 Ki = 328 nM T29741 CH6P3K 49837684 Ki = 520 nM T29741 C6ANT5 49837685 Ki = 565 nM T29741 C2MT0C 49837686 Ki = 235 nM T29741 C1X6GR 49837687 Ki = 428 nM T29741 CP3Z0G 49837783 Ki = 158 nM T29741 CFL8N3 49837784 Ki = 218 nM T29741 CQIL80 49837785 Ki = 515 nM T29741 CBZ74L 49837786 Ki = 259 nM T29741 CC4WF6 49837787 Ki = 236 nM T29741 CH8I0W 49837788 Ki = 387 nM T29741 CH28EJ 51035513 Ki = 144 nM T29741 C7OB2X 51035721 Ki = 72 nM T29741 C3AH5R 51035722 Ki = 76 nM T29741 CL96PR 51035723 Ki = 112 nM T29741 C56YLK 51035724 Ki = 101 nM T29741 CL2CN8 51035725 Ki = 87 nM T29741 C4LK5D 51035726 Ki = 103 nM T29741 C3H1VJ 51035928 Ki = 103 nM T29741 C91XOM 51035929 Ki = 111 nM T29741 C6U2YK 51035930 Ki = 116 nM T29741 C26PCE 51035931 Ki = 111 nM T29741 C42XGB 51035932 Ki = 142 nM T29741 CF8C6B 51036143 Ki = 93 nM T29741 C9B2SY 51036144 Ki = 131 nM T29741 CU04RE 51036146 Ki = 94 nM T29741 C58XAP 52940727 Ki > 30000 nM T29741 C31NIX 52942022 IC50 = 1640 nM T29741 CG3H5J 52942339 Ki = 47 nM T29741 CH0BQ4 52943153 IC50 = 1130 nM T29741 C76SDY 52943538 Ki = 398 nM T29741 CH0YN6 52945643 IC50 = 170 nM T29741 CIT05S 52946863 IC50 = 1400 nM T29741 C62QDZ 52948419 Ki = 240 nM T29741 CA9ME5 52949323 IC50 = 1070 nM T29741 CMX2N8 52949325 IC50 = 1300 nM T29741 C1DB7E 54703278 IC50 = 790 nM T29741 C1YQ7L 57395836 Ki = 67 nM T29741 C25RKI 57395837 Ki = 156 nM T29741 C8LUQ1 86301661 IC50 > 100000 nM T29741 CD0E3K 118718001 IC50 > 100000 nM T29741 C93NJU 118718002 IC50 > 100000 nM T29741 C8C5BD 118718020 IC50 > 100000 nM T29741 CT6K9C 118718021 IC50 > 100000 nM T29741 CJF9B1 118718025 IC50 > 100000 nM T29741 C49APK 118718026 IC50 > 100000 nM T29741 C8OJX0 118718040 IC50 > 100000 nM T29741 CST27I 118718052 IC50 > 100000 nM T29741 CI10BE 127043500 Ki = 6350 nM T29741 C6HFR0 127043501 Ki = 27700 nM T29741 CE4JF5 127043502 Ki = 24000 nM T29741 C3T8NG 127043677 Ki = 34600 nM T29741 C1O0RK 127043678 Ki = 2330 nM T29741 C2R5WP 127043810 Ki = 33800 nM T29741 CK0FU2 127044168 Ki = 37600 nM T29741 C7D9OK 127045101 Ki = 26400 nM T29741 CE1Z7H 127045569 Ki = 27000 nM T29741 CRHV36 127045603 Ki = 2390 nM T29741 CJ8YL1 127045604 Ki = 2630 nM T29741 CE0K6Z 127045605 Ki = 9310 nM T29741 COK81N 127045606 Ki = 840 nM T29741 CV1HQ8 127045607 Ki = 6830 nM T29741 CT5P4R 127045608 Ki = 2360 nM T29741 C9EA5L 135607310 IC50 = 1160 nM T29741 C2KQH1 135679117 IC50 = 910 nM T29741 CQEZ81 136002644 IC50 = 1020 nM T29741 C8RV0N 136002645 IC50 = 1000 nM T29741 C3CWN0 137443819 IC50 = 500 nM T29741 C8KRS9 137443821 IC50 = 27000 nM T29741 CCA9H3 137443825 IC50 = 3700 nM T29741 D00RIX 5280443 IC50 = 1130 nM T29741 D06UEP 17027464 Ki = 165 nM T29741 D0G3TK 5280863 IC50 = 1200 nM T19244 D00FGR 3599 IC50 > 100000 nM T19244 D00KHM 16362 IC50 > 30000 nM T19244 D00KVO 2082 IC50 > 30000 nM T19244 D00UVA 11556711 IC50 > 10000 nM T19244 D00YZD 54726191 IC50 > 100000 nM T19244 D01AXB 60835 IC50 = 29000 nM T19244 D01XNB 4594 Ki = 45000 nM T19244 D01ZII 2726 IC50 > 50000 nM T19244 D02HED 4748 IC50 = 21300 nM T19244 D02TJS 54676038 Ki = 600 nM T19244 D02VJP 25151504 IC50 > 25000 nM T19244 D03BLF 31307 IC50 > 50000 nM T19244 D03HFG 5324346 Ki = 8500 nM T19244 D03RTS 2662 IC50 = 10000 nM T19244 D03WEX 9966051 IC50 = 39000 nM T19244 D04JEE 4946 IC50 > 10000 nM T19244 D04NQI 2165 IC50 > 50000 nM T19244 D04OSE 4485 IC50 = 4080 nM T19244 D04XGT 31593 IC50 > 100000 nM T19244 D05CEU 941361 IC50 > 50000 nM T19244 D05DVP 5717 Ki = 2500 nM T19244 D05EAM 4735 IC50 > 25000 nM T19244 D05LBU 5472 IC50 = 31100 nM T19244 D05VIX 3463 IC50 = 9600 nM T19244 D06ABF 3957 IC50 > 30000 nM T19244 D06GDY 43815 IC50 > 30000 nM T19244 D06GKN 2099 IC50 < 10000 nM T19244 D06OIV 5505 Ki = 70000 nM T19244 D07ABV 468595 IC50 = 7200 nM T19244 D07ACT 5479530 IC50 > 50000 nM T19244 D07BPS 5359 Ki = 3700 nM T19244 D07BSQ 5994 Ki = 5500 nM T19244 D07ESC 11561674 IC50 > 10000 nM T19244 D07KSG 2733526 IC50 > 30000 nM T19244 D07UYO 441401 IC50 > 20000 nM T19244 D08QCJ 5430 Ki = 245000 nM T19244 D09GOS 2812 IC50 = 136 nM T19244 D09IPV 28417 IC50 = 1440 nM T19244 D09KTS 24821094 IC50 = 8500 nM T19244 D09LNI 3365 IC50 = 9210 nM T19244 D09SGV 25154714 IC50 = 59500 nM T19244 D0A4YE 5335 IC50 = 180 nM T19244 D0AZ8C 5213 Ki = 5000 nM T19244 D0C0SK 4993 Ki = 51500 nM T19244 D0C3SW 53465279 IC50 = 31200 nM T19244 D0D1AL 3559 IC50 > 30000 nM T19244 D0D4YZ 45375808 IC50 = 60000 nM T19244 D0D9FV 4601 IC50 > 30000 nM T19244 D0E3OF 54678486 Ki = 20000 nM T19244 D0E4DW 1775 Ki = 6000 nM T19244 D0F9BY 166548 IC50 > 17500 nM T19244 D0G4KG 3828 IC50 > 10000 nM T19244 D0H0KB 5070 IC50 > 25000 nM T19244 D0H0ND 54454 IC50 > 30000 nM T19244 D0I1FQ 54671008 IC50 > 50000 nM T19244 D0I2MK 4171 IC50 > 50000 nM T19244 D0K0TC 68617 IC50 > 50000 nM T19244 D0K8KX 5280343 IC50 = 10200 nM T19244 D0K9MY 11243969 IC50 > 50000 nM T19244 D0N3VR 71616 Ki = 2800 nM T19244 D0N6RF 65999 IC50 = 4780 nM T19244 D0NJ5H 11450633 IC50 < 10000 nM T19244 D0O3OS 104850 IC50 = 5.3 nM T19244 D0Q2PE 4539 IC50 > 50000 nM T19244 D0Q9EV 11965427 IC50 = 3000 nM T19244 D0R0FE 2520 IC50 > 30000 nM T19244 D0R1QE 3672 Ki = 50000 nM T19244 D0S5LO 25166913 IC50 > 30000 nM T19244 D0T0KA 4474 Ki = 280 nM T19244 D0T6WN 6451164 IC50 = 346 nM T19244 D0T8XB 44513473 IC50 > 10000 nM T19244 D0V7CF 5362440 IC50 > 30000 nM T19244 D0W7WC 16220172 IC50 > 20000 nM T19244 D0Y4JJ 2351 IC50 = 4310 nM T19244 D0Z1RV 135398737 IC50 = 21200 nM T19244 D0Z3DY 2333 Ki = 19 nM T19244 D0Z4EI 55245 IC50 = 4900 nM T19244 D0Z7KE 3784 IC50 = 3660 nM T19244 D0ZU9R 392622 IC50 = 4900 nM T19244 D00AUX 25230266 IC50 = 23000 nM T19244 D00DRL 44137946 IC50 = 1200 nM T19244 D00JFE 56941241 IC50 = 2200 nM T19244 D00RYA 16750271 IC50 > 10000 nM T19244 D00SWQ 10429242 IC50 = 22000 nM T19244 D01DDN 56950369 IC50 > 50000 nM T19244 D01LCC 17754438 IC50 = 5000 nM T19244 D02AAO 10368812 IC50 > 10000 nM T19244 D02ADM 31553 IC50 = 18000 nM T19244 D02AIN 122678117 IC50 > 20000 nM T19244 D02EEJ 6479267 IC50 = 13400 nM T19244 D02NNV 3038525 IC50 > 40000 nM T19244 D02QWY 24785538 IC50 = 23000 nM T19244 D02WFN 46207733 IC50 = 13300 nM T19244 D03AJU 44139752 IC50 > 10000 nM T19244 D03GNI 2166 IC50 = 75000 nM T19244 D03ISJ 135564632 IC50 > 50000 nM T19244 D03LWG 53235510 IC50 > 10000 nM T19244 D03MFQ 9996409 IC50 = 38000 nM T19244 D03MYO 15981237 IC50 = 22000 nM T19244 D03QHC 49856296 IC50 > 6000 nM T19244 D03SQT 68234908 IC50 > 100000 nM T19244 D03WNG 73051463 IC50 = 2000 nM T19244 D04MXN 56846693 IC50 > 10000 nM T19244 D04TNT 46851313 IC50 > 10000 nM T19244 D05LRD 59286554 IC50 > 30000 nM T19244 D05OMT 45142457 IC50 = 14730 nM T19244 D05PZB 135398495 IC50 > 10000 nM T19244 D05UYQ 15984937 IC50 > 100000 nM T19244 D06DMQ 59472121 IC50 > 30000 nM T19244 D06EPO 11192346 IC50 > 30000 nM T19244 D06TQR 76287260 IC50 = 11000 nM T19244 D06ZEO 54674461 IC50 > 50000 nM T19244 D07HZG 11516136 IC50 > 30000 nM T19244 D07OFM 46943432 IC50 >= 33000 nM T19244 D08AOZ 86582336 IC50 = 17100 nM T19244 D08PMW 9951995 IC50 = 1700 nM T19244 D08SCL 46190695 IC50 > 50000 nM T19244 D08VSQ 59336911 IC50 > 40000 nM T19244 D09DXX 71571306 IC50 > 100000 nM T19244 D09RII 71602803 IC50 = 8500 nM T19244 D09WYL 11634973 IC50 > 100000 nM T19244 D0A7ZK 56944144 IC50 > 20000 nM T19244 D0B5HF 44476893 IC50 > 50000 nM T19244 D0BM7M 11488320 IC50 > 10000 nM T19244 D0C5VQ 1548994 IC50 = 8200 nM T19244 D0C8DD 11552706 IC50 = 31622.78 nM T19244 D0C9PZ 91754484 IC50 = 23000 nM T19244 D0CB2B 23653789 IC50 = 30000 nM T19244 D0CG8S 71305058 IC50 > 25000 nM T19244 D0CW8S 71657619 IC50 > 50000 nM T19244 D0DH5X 44472635 IC50 > 100000 nM T19244 D0E0JO 117857370 EC50 > 100000 nM T19244 D0EB5N 25185057 IC50 > 25000 nM T19244 D0EY0A 42636350 IC50 > 30000 nM T19244 D0F4JK 11547499 IC50 > 30000 nM T19244 D0F4ZY 5311037 IC50 = 13000 nM T19244 D0F6YM 3035000 IC50 > 50000 nM T19244 D0G5XV 135565884 IC50 = 5700 nM T19244 D0G7UX 5284373 IC50 = 38800 nM T19244 D0G9AW 59473233 IC50 > 10000 nM T19244 D0GC5H 123879 IC50 = 15000 nM T19244 D0H9DA 54761306 IC50 > 10000 nM T19244 D0H9SX 6914657 IC50 = 3600 nM T19244 D0HE7C 134415769 IC50 > 10000 nM T19244 D0HS5V 11234052 IC50 > 40000 nM T19244 D0I2XM 3038500 IC50 = 24000 nM T19244 D0I3LO 91933883 IC50 > 20000 nM T19244 D0I3TU 45268455 IC50 = 5000 nM T19244 D0I4PW 60164925 IC50 > 50000 nM T19244 D0IA9Y 53472683 IC50 > 40000 nM T19244 D0IQ0Z 46885626 IC50 = 38000 nM T19244 D0IZ8X 90111638 IC50 > 51000 nM T19244 D0J1HB 23063810 IC50 > 100000 nM T19244 D0K1EG 11508736 IC50 > 100000 nM T19244 D0K4JQ 57339460 IC50 > 33000 nM T19244 D0K5HI 5311424 IC50 = 2000 nM T19244 D0K7FY 72703790 IC50 > 25000 nM T19244 D0L1GD 58282870 IC50 > 5000 nM T19244 D0L9KH 44623998 IC50 > 50000 nM T19244 D0L9QM 59568713 IC50 > 50000 nM T19244 D0LI1C 44469321 IC50 = 5420 nM T19244 D0LQ3L 77108121 IC50 = 25000 nM T19244 D0M4TJ 44219292 IC50 > 50000 nM T19244 D0M6BD 16719221 IC50 = 12000 nM T19244 D0M7CB 9919680 IC50 = 40000 nM T19244 D0M9RQ 11697697 IC50 > 21000 nM T19244 D0MR0B 54766013 IC50 > 10000 nM T19244 D0N5KS 154104 IC50 < 10000 nM T19244 D0N6NM 71721648 IC50 > 5600 nM T19244 D0N6SO 15983988 IC50 < 10000 nM T19244 D0O7QA 46840946 IC50 = 299 nM T19244 D0O9XN 11691484 IC50 = 5800 nM T19244 D0P0KN 16739650 IC50 > 25000 nM T19244 D0PN8H 46216796 IC50 > 5000 nM T19244 D0PW4N 6851740 IC50 > 25000 nM T19244 D0Q0AP 10409068 IC50 > 40000 nM T19244 D0Q7NB 10253143 IC50 > 100000 nM T19244 D0QR5G 2355 IC50 > 10000 nM T19244 D0R3VK 42642654 IC50 > 10000 nM T19244 D0RL4X 45270144 IC50 > 30000 nM T19244 D0S0EQ 9951066 IC50 = 14000 nM T19244 D0S1XX 134821691 IC50 > 40000 nM T19244 D0S2PD 42634627 IC50 > 30000 nM T19244 D0S5IR 86294073 IC50 > 30000 nM T19244 D0SG7B 49831257 IC50 > 70000 nM T19244 D0SP5V 49843471 IC50 > 50000 nM T19244 D0T3DO 9867758 IC50 = 25000 nM T19244 D0T4SG 11292191 IC50 > 10000 nM T19244 D0U4FF 10437018 IC50 = 12000 nM T19244 D0U7KH 86567195 IC50 > 5000 nM T19244 D0V9VG 51049968 IC50 >= 20000 nM T19244 D0VI4N 90409366 IC50 > 10000 nM T19244 D0W1US 1684 IC50 > 10000 nM T19244 D0W8XT 60663 IC50 = 28400 nM T19244 D0W9VW 11526696 IC50 = 66000 nM T19244 D0X7EG 11462174 IC50 > 30000 nM T19244 D0XD4I 118502708 IC50 > 30000 nM T19244 D0Y1NC 148198 IC50 = 120 nM T19244 D0Y7NA 49871007 IC50 > 25000 nM T19244 D0YB2Y 42641863 Ki > 30000 nM T19244 D0ZE1O 9949641 IC50 = 530 nM T19244 D0LF0O 135441202 IC50 > 40000 nM T19244 D03ZXG 118103874 IC50 = 5700 nM T19244 D08DMM 91799365 IC50 > 30000 nM T19244 D08SNH 71555922 IC50 = 3500 nM T19244 D0D3GL 137662068 IC50 > 40000 nM T19244 D0G2TX 46911228 IC50 > 5000 nM T19244 D0HG2S 86294663 IC50 = 4200 nM T19244 D0LI2I 118096900 IC50 > 30000 nM T19244 D0LU9X 74221950 IC50 > 50000 nM T19244 D0N6HP 91886057 IC50 = 5300 nM T19244 D0NJ9E 118096899 IC50 > 30000 nM T19244 D0QE8S 60197821 IC50 = 5400 nM T19244 D0TR9T 45256914 IC50 > 5000 nM T19244 D0W1XE 91827457 IC50 = 608 nM T19244 D0WR7B 122650373 IC50 > 30000 nM T19244 D03EZB 9864291 IC50 = 3600 nM T19244 D03YPJ 5163 IC50 > 100000 nM T19244 D04RLX 148201 IC50 = 7100 nM T19244 D04WCI 16220188 IC50 > 29000 nM T19244 D04YHW 11406590 IC50 > 40000 nM T19244 D05MCS 44473151 IC50 > 50 nM T19244 D06TGE 11226090 IC50 = 0.93 nM T19244 D06ZVC 10150497 IC50 > 500000 nM T19244 D07EBU 135565424 IC50 > 15000 nM T19244 D07GIB 11614352 IC50 > 50000 nM T19244 D08QHS 11296282 IC50 = 30 nM T19244 D08QTP 6478034 IC50 > 50000 nM T19244 D09EVZ 507806 IC50 = 30000 nM T19244 D09NBM 10417440 IC50 = 100000 nM T19244 D09VTB 71768520 IC50 >= 10000 nM T19244 D0A1NU 16049769 IC50 > 30000 nM T19244 D0B4TT 17747460 IC50 > 3000 nM T19244 D0B7SP 11292933 IC50 = 60000 nM T19244 D0G6SZ 3001322 IC50 > 30000 nM T19244 D0GE2F 53354790 IC50 = 4900 nM T19244 D0H9GQ 9795276 IC50 = 99000 nM T19244 D0IP6X 219077 IC50 = 11000 nM T19244 D0M4LF 23649325 IC50 = 3300 nM T19244 D0N8NK 11641563 IC50 > 10000 nM T19244 D0Q3ES 11705608 Ki = 100 nM T19244 D0R7GH 9833312 IC50 = 800 nM T19244 D0T0TZ 38409 Ki = 4300 nM T19244 D0Y2HR 2247 IC50 > 30000 nM T19244 D0YE2N 73214 IC50 > 20000 nM T19244 C4PZ9H 3444 IC50 = 8100 nM T19244 C9LCD8 3823 IC50 = 8940 nM T19244 C2KJI7 3883 IC50 = 19200 nM T19244 CN0WP7 15630 IC50 > 25000 nM T19244 C6GN7M 40692 IC50 > 30000 nM T19244 CK6VT0 60923 IC50 = 0.5 nM T19244 C2FVG0 64149 IC50 = 22000 nM T19244 CPW9G5 65126 Ki = 9200 nM T19244 CMLI08 68079 IC50 > 10000 nM T19244 C95JWC 68487 IC50 > 300000 nM T19244 CO0HB3 75473 Ki = 112000 nM T19244 C7SXL6 87152 IC50 > 25000 nM T19244 C2HFT4 91673 IC50 > 50000 nM T19244 CC0P7F 94378 IC50 = 9900 nM T19244 CZB67X 98608 IC50 > 10000 nM T19244 CHXZ93 101612 Ki = 6800 nM T19244 CH50RJ 104956 IC50 = 220 nM T19244 C0K7OY 108137 IC50 = 54000 nM T19244 CEP43C 122068 IC50 = 58000 nM T19244 C6QB9N 126266 IC50 = 50000 nM T19244 CZ67TG 145900 Ki = 35000 nM T19244 CM2H7V 152430 IC50 > 10000 nM T19244 CK8RD5 168114 IC50 = 6800 nM T19244 CJ34CF 168115 IC50 = 7500 nM T19244 CDB9P5 170922 IC50 > 25000 nM T19244 C1R6GB 189060 IC50 > 10000 nM T19244 CXE92M 234512 Ki = 125000 nM T19244 CAS18T 359052 IC50 > 30000 nM T19244 CDU5O6 421105 IC50 = 10000 nM T19244 CLD6J9 441074 Ki = 32000 nM T19244 COW92Q 447297 IC50 = 10000 nM T19244 CRH1D7 491206 IC50 = 2300 nM T19244 CKC8U4 507751 IC50 > 40000 nM T19244 CPXL01 507783 IC50 = 17000 nM T19244 CM40AT 507791 IC50 > 40000 nM T19244 C18QJF 515047 IC50 = 2600 nM T19244 CEN81S 515051 IC50 = 4500 nM T19244 CHX85A 515052 IC50 = 7400 nM T19244 C2Y4TD 577307 IC50 > 40000 nM T19244 C6R5XN 595145 IC50 = 99200 nM T19244 CVRM18 595254 Ki = 48200 nM T19244 CR98MZ 613528 IC50 > 30000 nM T19244 C4FC1N 626798 IC50 > 50000 nM T19244 CS5PK2 640180 IC50 = 67300 nM T19244 CTGL43 672443 IC50 = 50000 nM T19244 CGL5R1 683949 IC50 = 50000 nM T19244 CN5CJ7 688803 IC50 > 10000 nM T19244 C2AHB4 689051 IC50 > 10000 nM T19244 C74MRA 702869 IC50 = 6730 nM T19244 C6DJ3Y 741004 IC50 = 5980 nM T19244 C4V6EW 747770 IC50 > 30000 nM T19244 C4ZCO8 758155 Ki = 9940 nM T19244 CSUL21 780263 IC50 = 2540 nM T19244 CI43WJ 802727 IC50 > 10000 nM T19244 C3LM4S 821286 IC50 = 1600 nM T19244 C06WCN 827839 IC50 = 3250 nM T19244 CYKE37 863679 IC50 > 20000 nM T19244 CLJU94 877119 IC50 = 17600 nM T19244 C2TDG1 883547 IC50 > 40000 nM T19244 C2FPN5 936091 IC50 > 50000 nM T19244 CCKH57 969503 Ki = 6000 nM T19244 CMO9N5 970725 IC50 > 30000 nM T19244 CYF7O0 1121109 EC50 = 1584.89 nM T19244 C7ZAT5 1122589 EC50 = 3981.07 nM T19244 CI8G1R 1150344 Ki = 6000 nM T19244 CZG18E 1201554 Ki = 51500 nM T19244 CAZT67 1283333 IC50 = 6309.57 nM T19244 CV0Q3D 1302369 IC50 = 470 nM T19244 CU8G7F 1313100 EC50 = 251.19 nM T19244 C34YBF 1319308 EC50 = 2511.89 nM T19244 C5G4FA 1394668 IC50 > 30000 nM T19244 CMU8T3 1410239 IC50 = 4300 nM T19244 CP3F4T 1476707 IC50 > 50000 nM T19244 CW4YO2 1480806 IC50 = 39000 nM T19244 C0SLP9 1489193 IC50 = 15800 nM T19244 C0GE2X 1619763 IC50 = 3780 nM T19244 CC40IA 1909086 IC50 = 1000 nM T19244 C21HKV 1941609 IC50 = 410 nM T19244 C3LSW0 2088634 IC50 > 50000 nM T19244 CZL8R3 2187415 IC50 > 50000 nM T19244 CP53EV 2350190 IC50 = 1500 nM T19244 CQTY36 2650025 IC50 = 35800 nM T19244 CZY89U 2727594 IC50 = 4170 nM T19244 CD28JA 2735964 IC50 > 25000 nM T19244 C5T3HX 2748785 IC50 > 10000 nM T19244 C0ZI1F 2756534 IC50 = 26000 nM T19244 CT6P3F 2782903 IC50 = 7000 nM T19244 CF2N8O 2794167 IC50 > 30000 nM T19244 C07CXP 2805555 Ki = 17000 nM T19244 CTBC06 2941086 IC50 = 1258.93 nM T19244 C14NBG 3008866 IC50 = 5200 nM T19244 C4XNG5 3012020 IC50 = 10000 nM T19244 C6TO5V 3012027 IC50 = 6000 nM T19244 CCQI26 3012527 IC50 = 50000 nM T19244 CQ2SG0 3031421 IC50 > 20000 nM T19244 CAJQ53 3040177 Ki = 20900 nM T19244 C3GSR4 3114841 IC50 > 50000 nM T19244 C3F0GS 3120536 IC50 > 10000 nM T19244 CFPR85 3213696 IC50 > 5000 nM T19244 CZYR65 3261645 Ki = 20000 nM T19244 C2L9IF 3296768 IC50 = 21000 nM T19244 CI30FE 3463042 IC50 > 40000 nM T19244 C0BPL9 3707700 EC50 = 39810.72 nM T19244 CSW59H 3718258 IC50 = 10200 nM T19244 CXR4Y7 3811929 IC50 > 50000 nM T19244 CO23EI 3959338 IC50 > 20000 nM T19244 CEP9D5 4048115 IC50 > 50000 nM T19244 CG8A3J 4193543 IC50 = 4800 nM T19244 CIF8G9 4261503 IC50 = 11000 nM T19244 C1ZC4D 4384047 IC50 = 9730 nM T19244 CBSM52 4450788 IC50 = 500 nM T19244 C7RPL4 4450789 IC50 = 1300 nM T19244 CE0OD3 4652320 IC50 = 40000 nM T19244 CZO2E5 4674678 IC50 = 550 nM T19244 CBFV62 4817293 IC50 = 32700 nM T19244 CJ8PL6 4840815 IC50 = 43000 nM T19244 C7CNQ4 5201490 IC50 > 50000 nM T19244 CZM7D8 5281794 IC50 = 3300 nM T19244 C14OIP 5282539 IC50 = 500 nM T19244 CAMH93 5282542 IC50 = 2600 nM T19244 CO16PV 5282545 IC50 = 16000 nM T19244 C6C0UY 5282549 IC50 = 1400 nM T19244 CA5D1J 5289110 IC50 > 20000 nM T19244 CZ09MD 5299617 IC50 = 2200 nM T19244 CMBL90 5300578 IC50 > 20000 nM T19244 CA7UL5 5329333 IC50 > 50000 nM T19244 COQ41S 5329336 IC50 > 100000 nM T19244 COJI90 5338258 IC50 > 10000 nM T19244 CWFP51 5338324 IC50 > 10000 nM T19244 C5Z0HQ 5355549 IC50 > 20000 nM T19244 C7IKS9 5470829 IC50 = 2800 nM T19244 C3Q2XB 5495793 IC50 = 7900 nM T19244 C0ZAM9 5495818 IC50 > 40000 nM T19244 CH3GQ9 5708672 IC50 = 21300 nM T19244 CPT10H 5717399 IC50 > 20000 nM T19244 C21EJH 5717404 IC50 > 20000 nM T19244 CE9KZ5 5720628 IC50 > 20000 nM T19244 CJMQ48 5737900 IC50 > 20000 nM T19244 CSH9C1 5787676 IC50 > 20000 nM T19244 CMWC08 5837372 IC50 > 10000 nM T19244 CAJK62 5859537 IC50 > 20000 nM T19244 CX23PO 6020016 IC50 > 10000 nM T19244 C2V8QP 6174007 IC50 > 20000 nM T19244 CTG9I2 6258621 IC50 > 20000 nM T19244 CR8P9W 6262995 IC50 > 10000 nM T19244 CA74LD 6320546 IC50 > 30000 nM T19244 CY2A8V 6347538 Ki = 3300 nM T19244 CGJ16S 6436013 IC50 > 5000 nM T19244 CB75NI 6479949 IC50 > 30000 nM T19244 C09BQE 6479956 IC50 = 11500 nM T19244 CEL6U1 6479971 IC50 = 4000 nM T19244 CC6U7A 6493950 IC50 < 1000 nM T19244 CN0VB3 6914627 IC50 > 30000 nM T19244 C80XWJ 6914629 IC50 > 30000 nM T19244 C0QCK1 6918455 IC50 > 100000 nM T19244 CP8T7C 7017202 IC50 = 20000 nM T19244 C48OIX 7074967 Ki = 172000 nM T19244 CWX15G 7514880 IC50 > 20000 nM T19244 CJH57U 8854335 IC50 > 20000 nM T19244 C2W6PI 8867347 IC50 > 15000 nM T19244 C24MJV 9554928 IC50 = 1200 nM T19244 C32HVW 9554933 IC50 = 1400 nM T19244 CA15IT 9796590 IC50 > 30000 nM T19244 CUGX54 9797385 IC50 = 6500 nM T19244 CVZG73 9799417 IC50 = 80800 nM T19244 C5KZ9F 9805776 IC50 = 13000 nM T19244 CMIW83 9812710 IC50 > 30000 nM T19244 CR8ET5 9814387 IC50 = 40000 nM T19244 CFW74D 9815391 IC50 = 30000 nM T19244 CTN13P 9820134 IC50 = 52000 nM T19244 C1E2DV 9826083 IC50 > 2000 nM T19244 C3NO4W 9828630 IC50 = 1 nM T19244 C0UDC8 9839359 IC50 = 50000 nM T19244 C9IV7J 9844175 IC50 = 5700 nM T19244 CL79YZ 9858476 IC50 = 12000 nM T19244 C5O0RC 9866503 IC50 = 3900 nM T19244 CI6V2U 9870337 IC50 = 5900 nM T19244 CQ4LC2 9872676 IC50 = 3000 nM T19244 CTZP28 9875352 IC50 = 410 nM T19244 CBF9T3 9879532 IC50 = 31000 nM T19244 C8XNM3 9887837 Ki = 2200 nM T19244 CJW1P5 9888494 IC50 = 35000 nM T19244 C9C8JK 9890681 IC50 = 17000 nM T19244 CYHQ45 9906855 Ki = 36000 nM T19244 CUW29B 9908035 Ki = 64000 nM T19244 CJEP97 9908807 IC50 = 5470 nM T19244 C4B2QY 9913339 IC50 > 20000 nM T19244 C29WVT 9923385 IC50 > 25000 nM T19244 CFC48H 9940105 IC50 = 83900 nM T19244 CEB1I2 9945500 IC50 > 25000 nM T19244 CVYB74 9956808 IC50 = 3900 nM T19244 CNJ81W 9959174 IC50 = 9100 nM T19244 C74GQW 9960211 IC50 = 3600 nM T19244 CKLH03 9967123 IC50 = 12000 nM T19244 C8RD1Y 9980809 IC50 = 2900 nM T19244 CJOV70 9983904 IC50 = 14000 nM T19244 CGEJ24 9985625 IC50 = 5800 nM T19244 C98KZE 10002960 IC50 = 8400 nM T19244 C8F5KS 10005210 IC50 = 15000 nM T19244 C26QHZ 10005638 IC50 > 2000 nM T19244 CCD24K 10007859 IC50 >= 18000 nM T19244 CZ39MP 10020475 IC50 = 800 nM T19244 C45TBJ 10023245 IC50 = 5200 nM T19244 CW2X8U 10023735 IC50 = 1100 nM T19244 C5TRX2 10025406 IC50 = 8000 nM T19244 CA06TQ 10028888 IC50 > 100000 nM T19244 C1WH8Q 10042344 IC50 > 40000 nM T19244 CL58VA 10045582 IC50 = 60000 nM T19244 CGNA89 10045603 IC50 = 3000 nM T19244 C4SON9 10046844 IC50 = 1900 nM T19244 CPI2Q0 10049358 IC50 = 13000 nM T19244 CMSK43 10051746 IC50 = 15000 nM T19244 C4H6ZM 10063036 Ki = 6000 nM T19244 CSOR04 10070428 IC50 = 18000 nM T19244 C5B4HJ 10071498 IC50 = 75000 nM T19244 CVE2T1 10076176 IC50 > 10000 nM T19244 CR01QE 10076802 IC50 = 670 nM T19244 CF2ZS1 10099858 IC50 = 3500 nM T19244 CEA01V 10108128 IC50 = 33200 nM T19244 C3E4UM 10120032 IC50 = 600 nM T19244 CC2YT5 10122981 IC50 > 30000 nM T19244 C6HR7P 10130125 IC50 = 17000 nM T19244 C47RHT 10130685 IC50 = 300 nM T19244 CD75GU 10131619 IC50 > 10000 nM T19244 CP64RT 10134089 IC50 > 10000 nM T19244 CXS21P 10142377 IC50 = 9100 nM T19244 C2YZ4H 10144464 IC50 = 6400 nM T19244 CZG5Y6 10145190 IC50 = 700 nM T19244 C4F9HJ 10145470 IC50 = 4500 nM T19244 CR6H9Y 10146899 IC50 = 5500 nM T19244 C46EOS 10151840 IC50 = 5000 nM T19244 C0O2NM 10153212 IC50 = 2000 nM T19244 COFT51 10154555 IC50 = 1440 nM T19244 CQO8H3 10157813 IC50 = 30000 nM T19244 CLT63F 10166543 IC50 > 50000 nM T19244 C4NP8U 10167862 IC50 = 200 nM T19244 C8V2PN 10168172 IC50 = 200 nM T19244 CP6Q1W 10173403 IC50 = 45000 nM T19244 C73DEB 10181405 IC50 = 17000 nM T19244 C6OH0I 10184529 IC50 = 17000 nM T19244 CFUO45 10184774 IC50 = 15000 nM T19244 CJ1O9P 10185917 IC50 = 830 nM T19244 CYO0N7 10187078 IC50 = 3600 nM T19244 CKX0P3 10189203 IC50 = 11400 nM T19244 CEDW91 10190506 IC50 = 27300 nM T19244 CA4N2V 10198034 IC50 = 11000 nM T19244 CM0F5B 10198293 IC50 = 19600 nM T19244 C6JHB3 10210431 IC50 = 4600 nM T19244 CGMH76 10211390 IC50 = 3900 nM T19244 C8DWX5 10219789 IC50 = 35000 nM T19244 CX32UD 10223809 IC50 > 100000 nM T19244 CV5X8A 10224181 IC50 > 2500 nM T19244 C4JN9U 10224745 IC50 > 50000 nM T19244 C3FN5E 10226546 IC50 = 23000 nM T19244 C8DRL3 10232061 IC50 = 6900 nM T19244 C1B7ZE 10233723 IC50 = 48800 nM T19244 CK3Q4T 10245060 Ki = 100 nM T19244 C6UWX1 10254542 IC50 = 580 nM T19244 C3OE5Z 10257392 IC50 = 650 nM T19244 C4KU1Y 10268204 IC50 > 25000 nM T19244 CU1ZW4 10268255 IC50 = 500 nM T19244 C2EO1A 10273854 IC50 = 9000 nM T19244 CE9ID0 10280944 IC50 = 5500 nM T19244 C5T9IR 10282859 IC50 = 3800 nM T19244 CWOR29 10283706 IC50 > 30000 nM T19244 CO38FQ 10283896 IC50 = 28000 nM T19244 C16MNJ 10284289 IC50 < 1000 nM T19244 CO2LT5 10286610 IC50 = 24200 nM T19244 CD3BM8 10289976 IC50 = 7000 nM T19244 C7C5FN 10294289 IC50 < 1000 nM T19244 CE4Y7G 10294290 IC50 = 12800 nM T19244 C3FL9K 10295633 IC50 > 2000 nM T19244 C90DYG 10297996 IC50 = 59000 nM T19244 CO0P4F 10301330 IC50 = 5900 nM T19244 C9C3KH 10305705 IC50 = 19700 nM T19244 CAU47H 10305883 IC50 = 33000 nM T19244 CHOT95 10312127 IC50 = 14000 nM T19244 C6ITS2 10313487 IC50 > 100000 nM T19244 CZ18PL 10316203 IC50 >= 90000 nM T19244 C8F1LK 10318708 IC50 = 6000 nM T19244 C27TCH 10319351 IC50 = 12000 nM T19244 CT1XJ3 10323760 IC50 = 1600 nM T19244 CM46XO 10327211 IC50 = 6900 nM T19244 C7AY2L 10337564 IC50 = 5000 nM T19244 C4AJ0X 10341839 IC50 > 100000 nM T19244 CFXA48 10343679 IC50 > 25000 nM T19244 CJ7YZ9 10345293 IC50 = 1700 nM T19244 CW50TU 10345610 IC50 > 30000 nM T19244 C0OP5K 10347566 IC50 = 3200 nM T19244 CQVP17 10347783 IC50 = 15000 nM T19244 CH38EM 10353296 IC50 = 8000 nM T19244 CE19XH 10362365 IC50 = 16000 nM T19244 CW9P2U 10364379 IC50 = 9000 nM T19244 C4VJB9 10364714 IC50 = 36000 nM T19244 CN2ZH1 10364928 IC50 = 20000 nM T19244 C68MRW 10367597 IC50 = 7200 nM T19244 CDA5F7 10369999 IC50 = 230 nM T19244 C4A5SP 10379988 IC50 > 10000 nM T19244 C9QEO8 10386398 IC50 = 110 nM T19244 C3UM5T 10388098 IC50 = 26000 nM T19244 C07XHY 10388612 IC50 = 3600 nM T19244 CA8B5T 10390073 IC50 > 2000 nM T19244 CU6Q5V 10390387 IC50 = 730 nM T19244 CJQV19 10391684 IC50 = 2200 nM T19244 C4H8ZC 10392194 IC50 = 38 nM T19244 CWK4O1 10406239 IC50 >= 5000 nM T19244 C8K7VS 10410589 IC50 = 37000 nM T19244 CR1YG5 10415353 IC50 > 100000 nM T19244 CBN4H0 10415698 IC50 = 410 nM T19244 C97LHV 10454092 IC50 = 900 nM T19244 C8DWH6 10456892 IC50 > 30000 nM T19244 C25FVM 10457343 IC50 > 100000 nM T19244 C1H5RP 10458842 IC50 > 10000 nM T19244 CNGF26 10476287 IC50 = 4000 nM T19244 CXA0Q9 10479990 IC50 = 9800 nM T19244 CXB9T0 10480864 IC50 = 1600 nM T19244 C84ZBK 10481134 IC50 = 4000 nM T19244 CGXY36 10482372 IC50 = 2300 nM T19244 CWI7U5 10497417 Ki = 2400 nM T19244 C8TPU0 10510985 Ki = 6300 nM T19244 CKBU57 10519399 Ki = 6000 nM T19244 CBOL80 10612767 Ki = 18000 nM T19244 C2ONR8 10617103 Ki = 400 nM T19244 C6UX4J 10633725 IC50 > 10000 nM T19244 CD2JL5 10637940 Ki = 7000 nM T19244 CJPW17 10654534 Ki > 400000 nM T19244 CQSJ50 10692619 IC50 = 37700 nM T19244 CA82YQ 10704488 IC50 > 20000 nM T19244 C0ZD2I 10709273 Ki = 2000 nM T19244 CR4BW5 10760152 IC50 = 28313919.96 nM T19244 C9SWF5 10791993 IC50 = 54954087.39 nM T19244 CHMR42 10801437 Ki = 3000 nM T19244 CQTB48 10826603 Ki = 48000 nM T19244 CJ4D8N 10829073 Ki = 25000 nM T19244 CXK63D 10829689 IC50 = 62800 nM T19244 C0DM8R 10833710 Ki = 37000 nM T19244 CNS12Z 10850049 Ki = 18000 nM T19244 CG1L6V 10861208 IC50 = 55000 nM T19244 CJQ6E2 10861641 IC50 > 100000 nM T19244 CBK06L 10861643 IC50 = 492000 nM T19244 CK95RM 10894740 IC50 = 55000 nM T19244 CH0Z6X 10895263 IC50 > 200000 nM T19244 CZS9Q5 10899427 IC50 = 55200 nM T19244 C8Q9MI 10916150 IC50 = 12000 nM T19244 CC8K0J 10925491 IC50 = 100000 nM T19244 C35ZVX 10938153 IC50 = 80000 nM T19244 CI87GM 10938696 IC50 = 4000 nM T19244 CIG05D 10948187 IC50 > 200000 nM T19244 C4D9MR 10950401 IC50 = 12000 nM T19244 CE2O7T 11013215 IC50 = 1000 nM T19244 C6D2WT 11046887 IC50 = 50000 nM T19244 C1INT8 11070834 IC50 = 28000 nM T19244 CGT39L 11078396 IC50 = 90000 nM T19244 C34FLK 11100382 IC50 = 80000 nM T19244 CQ8DF3 11103028 IC50 = 15000 nM T19244 CFA1J0 11123454 IC50 = 20000 nM T19244 CH61UW 11128957 IC50 > 20000 nM T19244 CUB7H2 11133137 IC50 = 10000 nM T19244 CW1Q6S 11148656 IC50 < 46 nM T19244 CCD91J 11148936 IC50 = 10200 nM T19244 CXT8Y2 11151568 IC50 < 10000 nM T19244 CB47FY 11154357 IC50 = 43000 nM T19244 CFS2N7 11154496 IC50 = 10000 nM T19244 C5K4PC 11160258 IC50 = 7740 nM T19244 C1A8HL 11171679 Ki = 111000 nM T19244 CP1EI3 11172276 IC50 = 6880 nM T19244 C0EC8V 11181988 Ki = 145000 nM T19244 CRU5Y3 11183547 IC50 = 6090 nM T19244 CY57GR 11187635 IC50 = 8790 nM T19244 C0XCD3 11195292 IC50 = 27200 nM T19244 C7F6CE 11195591 IC50 = 6480 nM T19244 CHM83A 11199490 IC50 = 18400 nM T19244 CL9BN8 11202851 IC50 = 37660 nM T19244 C1XR3I 11206290 Ki = 4500 nM T19244 CJ1O6V 11207072 IC50 = 26900 nM T19244 CV1SD9 11208566 IC50 > 10000 nM T19244 CE0WA5 11211840 IC50 = 7300 nM T19244 C4O3QM 11218177 IC50 = 25000 nM T19244 CI2SN0 11222420 IC50 = 600 nM T19244 CEW9L6 11228293 IC50 > 5000 nM T19244 CMHY80 11229234 Ki = 38100 nM T19244 CA71OC 11235004 IC50 > 100000 nM T19244 C9WY6K 11235389 IC50 > 50000 nM T19244 C6D3UR 11237434 IC50 > 30000 nM T19244 C8IQ7N 11247557 IC50 = 16000 nM T19244 CLR09Q 11253245 IC50 = 5220 nM T19244 C7KU1G 11264664 IC50 > 46 nM T19244 C0XN7E 11272006 IC50 = 50680 nM T19244 C9W2NY 11274374 IC50 > 10000 nM T19244 C9W4KE 11275964 IC50 > 100000 nM T19244 CBEW43 11308052 IC50 = 15000 nM T19244 CF5YS9 11310529 Ki = 103000 nM T19244 CB7YS1 11315814 IC50 > 5000 nM T19244 C8S4FU 11317045 IC50 > 29100 nM T19244 CO8B7R 11317439 IC50 > 25000 nM T19244 CMQD35 11321674 Ki = 33900 nM T19244 C7WA0E 11322127 IC50 < 46 nM T19244 CY9KM7 11322128 IC50 = 26400 nM T19244 CT6CH4 11322177 IC50 = 8700 nM T19244 CW01KR 11322201 IC50 = 8180 nM T19244 CU72EY 11344157 Ki = 39700 nM T19244 CPK71M 11345209 IC50 = 36800 nM T19244 C5FG8X 11355925 IC50 = 398000 nM T19244 C7I4FX 11363702 IC50 > 10000 nM T19244 C8N0GX 11368215 IC50 = 88 nM T19244 C1RD9J 11369883 Ki = 40 nM T19244 CC0L7O 11377200 IC50 = 28000 nM T19244 C1BOK3 11378800 Ki = 61500 nM T19244 C0YO8L 11378954 IC50 = 43300 nM T19244 CD82VI 11379226 IC50 = 17800 nM T19244 CD68AR 11380674 IC50 < 50 nM T19244 CZIC23 11389737 IC50 > 400000 nM T19244 CYL06Q 11389927 IC50 > 400000 nM T19244 C9AOM3 11397017 IC50 > 10000 nM T19244 CLR3W7 11424804 IC50 < 46 nM T19244 CUSQ84 11430331 IC50 = 24000 nM T19244 C3CU1H 11450354 IC50 > 40000 nM T19244 CE42DM 11453673 IC50 = 2800 nM T19244 CPIH90 11458616 IC50 = 2800 nM T19244 CIDT15 11464169 IC50 = 4300 nM T19244 CR4N5I 11465834 IC50 = 49000 nM T19244 CW57BU 11480732 IC50 = 75200 nM T19244 COC7Q9 11488952 IC50 = 3500 nM T19244 CW3YO5 11494768 IC50 > 50000 nM T19244 CL17QT 11497455 IC50 > 10000 nM T19244 CTYJ07 11501580 IC50 = 42000 nM T19244 CL4J9A 11501698 IC50 = 1500 nM T19244 CR5I6K 11503692 IC50 = 5300 nM T19244 CFSH67 11504490 IC50 > 10000 nM T19244 C97WGN 11505187 IC50 > 10000 nM T19244 CQ6IU7 11509269 IC50 > 10000 nM T19244 C2T8YD 11511361 IC50 > 10000 nM T19244 CP8B7T 11511719 IC50 > 10000 nM T19244 C0SN2O 11515728 IC50 > 10000 nM T19244 COTH53 11516139 IC50 = 17000 nM T19244 C6ZG5T 11516324 IC50 = 9200 nM T19244 C6CV5S 11516424 IC50 = 22000 nM T19244 CVNP35 11517292 IC50 > 10000 nM T19244 CG3BZ9 11517980 IC50 = 8000 nM T19244 CUDR26 11518018 IC50 = 1800 nM T19244 CX4MA8 11519486 IC50 > 40000 nM T19244 CY47AQ 11519784 IC50 > 10000 nM T19244 CVO7T9 11522969 IC50 > 10000 nM T19244 CVPX30 11523521 IC50 = 7000 nM T19244 C4GLJ5 11524843 IC50 > 10000 nM T19244 CF3OE8 11525105 IC50 = 2500 nM T19244 CQ3TO7 11526741 IC50 > 10000 nM T19244 C7HNP0 11526745 IC50 > 100000 nM T19244 C0BF5R 11527661 IC50 > 25000 nM T19244 C75FPD 11529874 IC50 > 3000 nM T19244 C4Q8VK 11533340 IC50 > 10000 nM T19244 CR92GA 11537005 IC50 = 120 nM T19244 CF2OM8 11539410 IC50 = 14000 nM T19244 CFS7T8 11540675 IC50 = 5380 nM T19244 C2C7YA 11541635 IC50 = 2000 nM T19244 C3VP9T 11544537 IC50 > 10000 nM T19244 CD1YT8 11547169 IC50 = 3300 nM T19244 CP4HI9 11547703 IC50 = 6000 nM T19244 C7IOJ0 11548023 IC50 = 2500 nM T19244 CRZ7H2 11556677 IC50 = 5500 nM T19244 CQJ54M 11560300 IC50 < 400 nM T19244 C84NIF 11566130 IC50 > 10000 nM T19244 CDFU34 11566489 IC50 > 10000 nM T19244 CB59HM 11570626 IC50 = 14000 nM T19244 C4IX6W 11573549 IC50 > 10000 nM T19244 C7COV1 11576252 IC50 = 3000 nM T19244 CTVX46 11576269 IC50 > 10000 nM T19244 CFP36L 11576510 IC50 = 740 nM T19244 CR75FZ 11577204 IC50 < 300 nM T19244 CVX6K7 11580514 IC50 > 10000 nM T19244 C3YXZ7 11582291 IC50 = 15000 nM T19244 CFZ1Q5 11584681 IC50 = 39000 nM T19244 CFU15B 11588489 IC50 = 216000 nM T19244 C1HG4A 11591164 IC50 = 2000 nM T19244 C2Q8FI 11592021 IC50 = 6700 nM T19244 C06OQG 11598554 IC50 > 33000 nM T19244 CHU90R 11598626 IC50 > 8000 nM T19244 CP56DO 11599295 IC50 > 10000 nM T19244 CR37EA 11602469 IC50 = 4700 nM T19244 C4ALS8 11602549 IC50 = 28000 nM T19244 C15TEH 11604449 IC50 > 10000 nM T19244 CKJ4G0 11606814 IC50 = 330 nM T19244 CPH40V 11607042 IC50 = 13500 nM T19244 CH7P9Z 11608743 IC50 > 30000 nM T19244 C7ENB2 11609939 IC50 = 89000 nM T19244 C2M8HZ 11610353 IC50 > 50000 nM T19244 C8J3BY 11610363 IC50 = 4200 nM T19244 CKXH63 11610910 IC50 > 12000 nM T19244 CM7LS0 11612187 IC50 = 21000 nM T19244 C6LUG4 11612700 IC50 = 540 nM T19244 C5JZ6R 11615459 IC50 > 40000 nM T19244 C0R1SW 11617480 IC50 = 1600 nM T19244 CW0ZM6 11619260 IC50 > 50000 nM T19244 CMHG86 11620404 IC50 = 4877 nM T19244 CSM62L 11626920 IC50 = 700 nM T19244 CGX96V 11626927 IC50 < 50118.72 nM T19244 C3CP2G 11627368 IC50 > 10000 nM T19244 C9L5VD 11631813 IC50 = 43000 nM T19244 CM1DR9 11632375 IC50 = 12000 nM T19244 CYL45U 11634544 IC50 > 10000 nM T19244 CSM83G 11634807 IC50 = 4700 nM T19244 CCP69D 11638499 IC50 > 10000 nM T19244 CRT09O 11638500 IC50 > 10000 nM T19244 CF7X3A 11640317 IC50 = 6500 nM T19244 CT4BE7 11641076 IC50 = 26000 nM T19244 CTXG50 11642625 IC50 > 10000 nM T19244 CPV95E 11646179 IC50 < 140 nM T19244 C6Y4HR 11647548 IC50 > 30000 nM T19244 CYV4G6 11648801 IC50 = 4100 nM T19244 CMB6F9 11653874 IC50 = 40000 nM T19244 CB7P8J 11655677 IC50 = 19000 nM T19244 CX7FR8 11655728 IC50 > 9000 nM T19244 C51UDK 11667741 IC50 > 10000 nM T19244 CXJ17M 11669364 IC50 = 16000 nM T19244 CYM68U 11670135 IC50 = 6920 nM T19244 CIUJ01 11670392 IC50 = 2000 nM T19244 C0V7SU 11675388 IC50 = 1000 nM T19244 CULF07 11676720 IC50 = 4000 nM T19244 CFYQ85 11677212 IC50 = 1200 nM T19244 C72BNQ 11682521 IC50 > 50000 nM T19244 CW4U3H 11688520 IC50 > 10000 nM T19244 C3WBU8 11689242 IC50 = 4700 nM T19244 CH96LS 11692059 IC50 > 10000 nM T19244 CYB9E3 11692359 IC50 = 30000 nM T19244 C9CM2R 11695689 IC50 = 15000 nM T19244 COH3C4 11697546 IC50 = 640 nM T19244 C3XYS6 11698194 IC50 = 2000 nM T19244 C9J1QT 11698844 IC50 = 2800 nM T19244 C5ECV1 11699447 IC50 > 35000 nM T19244 C4DJ1V 11699804 IC50 > 10000 nM T19244 CO3U4B 11705008 IC50 = 8000 nM T19244 C7YHW1 11705018 IC50 = 8400 nM T19244 C73UBS 11709395 IC50 = 19000 nM T19244 CL4DS1 11709762 IC50 > 10000 nM T19244 CK4I6J 11710700 IC50 > 40000 nM T19244 C5FZ1J 11710873 IC50 = 35000 nM T19244 CHK5I2 11712756 IC50 > 9000 nM T19244 CN5UX7 11713409 IC50 = 21000 nM T19244 CL5S9K 11719046 IC50 > 5000 nM T19244 CZY05V 11719421 IC50 > 100000 nM T19244 CD9A0J 11720104 IC50 = 4100 nM T19244 CX9VH0 11720815 IC50 > 10000 nM T19244 CC05TM 11732429 IC50 = 50000 nM T19244 C0Z5JS 11740023 IC50 = 16000 nM T19244 CNJD24 11741843 IC50 = 630 nM T19244 CG0YB2 11751828 IC50 > 10000 nM T19244 CC92YE 11755033 IC50 > 100000 nM T19244 C58DMZ 11757696 IC50 = 550 nM T19244 CE19RO 11760273 IC50 = 26000 nM T19244 C8D7BS 11771234 IC50 > 20000 nM T19244 CB36OJ 11771503 IC50 > 40000 nM T19244 C6TS4D 11773824 IC50 > 5000 nM T19244 C6A1LM 11786814 IC50 = 40000 nM T19244 CN8CP5 11817019 IC50 = 7520 nM T19244 CS7W2V 11848793 IC50 = 8000 nM T19244 CI6JQ5 11855008 IC50 = 129000 nM T19244 CL1FX0 11947758 IC50 > 30000 nM T19244 CK2EZ6 11962967 IC50 = 17000 nM T19244 CH26TZ 11963255 IC50 = 16000 nM T19244 C8P9GD 11966041 IC50 > 10000 nM T19244 CYEN98 11977494 IC50 = 44000 nM T19244 CN5W3V 11978858 IC50 = 11300 nM T19244 CW8T4V 11978859 IC50 = 15300 nM T19244 CM07WK 11993787 IC50 = 2400 nM T19244 C1T8XZ 11993865 Ki = 14500 nM T19244 CBZ83S 11993868 Ki > 400000 nM T19244 C7A1EZ 11993870 Ki = 24200 nM T19244 C4XP2N 11993872 Ki = 2900 nM T19244 CWT0S3 11993875 Ki = 500 nM T19244 CR4YS2 11996303 IC50 = 9000 nM T19244 C7D1AY 11996304 IC50 = 2000 nM T19244 C1A2IB 12001199 IC50 > 100000 nM T19244 C9RX1L 12108566 IC50 = 30000 nM T19244 CO3HN1 13163256 IC50 = 79000 nM T19244 C1W2YO 13336341 Ki = 23610 nM T19244 CO4H3X 13427248 Ki = 1500 nM T19244 C9OJ8U 13427249 Ki = 20000 nM T19244 C6EPU4 13427251 Ki = 1100 nM T19244 CPBT26 13427253 Ki = 2400 nM T19244 C7I9PF 13557523 Ki > 400000 nM T19244 C0FY4P 13615899 IC50 > 20000 nM T19244 CO76XB 13927314 IC50 = 16000 nM T19244 C1G0EZ 13957609 IC50 = 6970 nM T19244 CIF90V 14434140 IC50 > 20000 nM T19244 C3YRU7 15295578 IC50 = 600 nM T19244 C7X3CQ 15604497 IC50 = 1584.89 nM T19244 CT4RL1 15778480 IC50 = 98200 nM T19244 CBE59I 15940927 IC50 = 40300 nM T19244 C08NEU 15945881 IC50 > 10000 nM T19244 C79VQK 15950271 IC50 > 10000 nM T19244 C3BI9R 15951010 IC50 > 10000 nM T19244 CWH1A8 15951076 IC50 > 10000 nM T19244 C2ZYA6 15951338 IC50 > 100000 nM T19244 C1Q8IV 15951410 IC50 = 21500 nM T19244 CUI7P4 15955613 IC50 < 1000 nM T19244 C3W8ZL 15981007 IC50 > 50000 nM T19244 CW6S0H 15981486 IC50 = 9000 nM T19244 C7SN1C 15983053 IC50 = 7100 nM T19244 CS97JR 15983175 IC50 > 20000 nM T19244 C0O5BA 15983546 IC50 > 50000 nM T19244 C83NXU 15983672 IC50 = 5900 nM T19244 C2D1KP 15983982 IC50 = 10400 nM T19244 CQJ7Y2 15985912 IC50 = 630.96 nM T19244 CPR25X 15986917 IC50 > 100000 nM T19244 C0DWJ8 15986929 IC50 > 100000 nM T19244 CR9FH7 15986930 IC50 = 12000 nM T19244 CEMJ79 15986931 IC50 = 12000 nM T19244 CX37OI 15986936 IC50 > 50000 nM T19244 C5KW3L 15987108 IC50 > 100000 nM T19244 CCL59Z 16007088 IC50 > 10000 nM T19244 C08CSK 16007091 IC50 > 18000 nM T19244 CG5A7W 16013152 IC50 = 990 nM T19244 CBMF65 16013184 IC50 = 21000 nM T19244 C6V4TG 16013186 IC50 = 45000 nM T19244 C20CRP 16040587 IC50 > 100000 nM T19244 C8ZP3G 16041292 IC50 > 100000 nM T19244 CDU1L0 16041411 IC50 > 60000 nM T19244 CMZU26 16043268 IC50 = 10500 nM T19244 C29KFG 16045493 IC50 = 10300 nM T19244 CQ9U1Y 16051921 IC50 = 62000 nM T19244 C30UFT 16066811 IC50 = 24500 nM T19244 CFK8J5 16068056 IC50 > 25000 nM T19244 CQRU95 16070337 IC50 = 25000 nM T19244 C8E6CH 16070448 IC50 > 25000 nM T19244 CTIQ90 16071896 IC50 > 25000 nM T19244 CX2GC6 16071897 IC50 > 25000 nM T19244 CL4ON2 16072021 IC50 = 5000 nM T19244 CJU50N 16072099 IC50 = 2080 nM T19244 C8D0KF 16099905 IC50 = 2000 nM T19244 C2FXW0 16099923 IC50 = 8200 nM T19244 C37LJV 16102853 IC50 > 50000 nM T19244 CEF3A0 16102867 IC50 = 8900 nM T19244 C91AZO 16102868 IC50 = 4700 nM T19244 CC24LB 16110489 IC50 > 10000 nM T19244 CHR8G4 16122633 IC50 > 10000 nM T19244 C0S1VK 16122818 IC50 > 40000 nM T19244 CFYL31 16122898 IC50 > 50000 nM T19244 C9G8TZ 16124598 IC50 = 21379.62 nM T19244 C0J6CH 16125372 IC50 = 7000 nM T19244 CMN0P3 16125681 IC50 = 4200 nM T19244 C4BYI2 16125682 IC50 = 7300 nM T19244 C8FLH6 16202152 IC50 = 10000 nM T19244 CWJZ50 16223655 IC50 = 9.1 nM T19244 CDG38L 16223656 IC50 > 10 nM T19244 C3O7HD 16223851 IC50 = 15.5 nM T19244 C0D9KR 16223854 IC50 = 26.9 nM T19244 C5L1QM 16224456 IC50 > 50 nM T19244 CTH6W4 16292141 IC50 > 25000 nM T19244 CQ3HO2 16309462 IC50 = 5800 nM T19244 C07CYO 16432973 Ki = 100 nM T19244 CVJ4O1 16654686 Ki > 300000 nM T19244 CY6D1F 16656782 IC50 = 11100 nM T19244 C6P4BX 16656803 IC50 > 25000 nM T19244 C7X0TS 16659334 IC50 > 30000 nM T19244 CIBY49 16661548 IC50 = 2400 nM T19244 C45KPZ 16661549 IC50 = 870 nM T19244 CH60SU 16661701 IC50 = 1700 nM T19244 CU9LS2 16661702 IC50 = 1100 nM T19244 CXL4Q3 16663122 IC50 = 500 nM T19244 CK4FJ8 16664733 IC50 = 5100 nM T19244 C1UY8J 16666386 IC50 = 7900 nM T19244 CH0Q9T 16678616 IC50 > 50000 nM T19244 C4FUO7 16678620 IC50 > 50000 nM T19244 CDY08B 16678725 IC50 > 50000 nM T19244 C1N8IL 16679518 IC50 > 50000 nM T19244 C0CF9G 16679612 IC50 > 50000 nM T19244 C8X6SN 16679614 IC50 > 50000 nM T19244 CH8A2G 16679616 IC50 > 50000 nM T19244 CBE9O8 16679617 IC50 > 50000 nM T19244 CQF5Y7 16679701 IC50 > 50000 nM T19244 CSK8N5 16679707 IC50 > 50000 nM T19244 CK9IU2 16718491 IC50 > 10000 nM T19244 CAPU50 16719554 IC50 = 10000 nM T19244 CN95DG 16719649 IC50 > 100000 nM T19244 C92NRU 16727109 IC50 > 40000 nM T19244 CG04RZ 16727123 IC50 = 1000 nM T19244 CAX2B7 16728787 IC50 = 3700 nM T19244 C0H8UN 16730109 IC50 > 40000 nM T19244 C9BC0L 16732000 IC50 > 40000 nM T19244 CHU72I 16738321 IC50 = 110 nM T19244 CN5GT7 16739030 IC50 = 1400 nM T19244 CBR95H 16739953 IC50 = 4400 nM T19244 CLY57P 16744597 IC50 > 40000 nM T19244 CA68OS 16744599 IC50 = 40000 nM T19244 CUI0X4 16744748 IC50 > 40000 nM T19244 CM3OV0 16745085 IC50 = 19000 nM T19244 C94MKR 16745086 IC50 = 40000 nM T19244 C5GY6N 16745241 IC50 = 15000 nM T19244 CW85LQ 16745311 IC50 = 96.8 nM T19244 CC4L1M 16747701 IC50 > 22000 nM T19244 C5DKZ8 16956771 IC50 > 11000 nM T19244 C9XS6P 17014937 Ki = 4060 nM T19244 CU42ZC 17244953 IC50 > 25000 nM T19244 C8D4PX 17408359 IC50 > 20000 nM T19244 CEV2A8 17605927 Ki = 15000 nM T19244 C8O3JV 17720407 Ki = 3470 nM T19244 C9C5TV 17751819 IC50 = 10000 nM T19244 C8TKD5 17754437 IC50 > 100000 nM T19244 CAJ0S2 17754557 EC50 > 50000 nM T19244 CH61IT 17754941 IC50 > 40000 nM T19244 CJK53H 17754942 IC50 > 40000 nM T19244 CHG32A 17755034 IC50 = 25000 nM T19244 C87WIK 18104758 IC50 > 50000 nM T19244 C4ZH0B 18274179 Ki = 1150 nM T19244 CF9TW8 18414685 IC50 = 8800 nM T19244 CG93TR 18440026 IC50 = 8000 nM T19244 C2HFY3 19553304 IC50 > 20000 nM T19244 CKH72O 20115797 IC50 = 50000 nM T19244 CR1K3H 20763282 IC50 = 42000 nM T19244 C8X0RI 20763372 IC50 = 17000 nM T19244 C8OHP4 20763385 IC50 = 19900 nM T19244 C6POY9 20763386 IC50 = 8800 nM T19244 CZBJ32 20763421 IC50 = 24000 nM T19244 C7OMR1 20763606 IC50 = 77000 nM T19244 C81JWV 20906619 IC50 = 3000 nM T19244 CHC4Q3 21064283 IC50 = 8800 nM T19244 C1CA6D 21070989 IC50 > 10000 nM T19244 CAW9T6 21105257 IC50 >= 24000 nM T19244 C6AU1N 21112865 IC50 = 14000 nM T19244 CTSG57 21112869 IC50 = 12000 nM T19244 C13HXO 21112870 IC50 = 5400 nM T19244 CY9B5M 21257907 IC50 = 1900 nM T19244 CWQ70U 21260391 IC50 = 12450 nM T19244 CO17PU 21635104 IC50 = 19952.62 nM T19244 CO6E2Z 21717336 IC50 = 16000 nM T19244 C7KIJ3 21717337 IC50 = 1500 nM T19244 CM1IF8 21914519 IC50 = 39810.72 nM T19244 CK4L1Y 21914620 IC50 = 31622.78 nM T19244 CZF82E 21914667 IC50 = 63095.73 nM T19244 CK8X7S 21956341 IC50 = 700 nM T19244 CO32YX 22254068 IC50 > 10000 nM T19244 C4YP8N 22431956 IC50 > 20000 nM T19244 C9N5XW 22520172 IC50 = 1700 nM T19244 C7J8HR 22965614 IC50 > 40000 nM T19244 C3TVL7 23501721 IC50 > 12500 nM T19244 CF81SW 23582412 IC50 > 100000 nM T19244 C9K1DY 23583191 IC50 > 100000 nM T19244 C0EJK3 23585071 IC50 = 5000 nM T19244 CW2R4M 23624283 IC50 > 100000 nM T19244 CQ29HW 23626128 IC50 > 20000 nM T19244 C0HA4Y 23626131 IC50 > 20000 nM T19244 C3Z6LM 23626132 IC50 > 20000 nM T19244 C2EXB1 23626439 IC50 > 20000 nM T19244 C7EK4A 23626924 IC50 > 20000 nM T19244 CW6OB1 23627212 IC50 > 10000 nM T19244 CWAT04 23630291 IC50 = 4000 nM T19244 CMQ6W7 23630305 IC50 > 10000 nM T19244 CHU29W 23635235 IC50 > 10000 nM T19244 CDL4G9 23645678 IC50 > 200000 nM T19244 C1AQ9P 23647882 IC50 > 30000 nM T19244 CTJ2P1 23647883 IC50 = 30000 nM T19244 CU6E5F 23647884 IC50 = 15000 nM T19244 C6NS9I 23647885 IC50 > 30000 nM T19244 CD9IC3 23647886 IC50 > 30000 nM T19244 CPX95O 23647887 IC50 = 4900 nM T19244 CK9D8P 23647888 IC50 = 8300 nM T19244 CX50BA 23647889 IC50 > 22000 nM T19244 C37JMS 23647890 IC50 = 12000 nM T19244 CJ97BQ 23647892 IC50 > 30000 nM T19244 CXP2G5 23647893 IC50 > 30000 nM T19244 C3JBX4 23647894 IC50 > 30000 nM T19244 CZ0QF1 23648867 IC50 > 30000 nM T19244 CR0VF4 23649212 IC50 = 2500 nM T19244 CK76FP 23649427 IC50 > 100 nM T19244 CAUC58 23649669 IC50 > 100000 nM T19244 CBZF78 23653563 IC50 = 3000 nM T19244 CG39XH 23654666 IC50 > 100 nM T19244 C6VSO8 23657438 IC50 = 5000 nM T19244 CFMX27 23658550 IC50 = 6800 nM T19244 CRW4V9 23663996 Ki = 7400 nM T19244 C5D3RZ 23683143 IC50 = 4800 nM T19244 C26ANU 23696680 IC50 = 15000 nM T19244 CASU54 23696973 IC50 = 8000 nM T19244 CS5E6J 23729988 IC50 > 900000 nM T19244 C93CGU 23904404 Ki = 5930 nM T19244 CK2Q5J 24180592 IC50 > 10000 nM T19244 C9R1PK 24180717 IC50 > 20000 nM T19244 CZ03FI 24649020 IC50 > 50000 nM T19244 CIAV47 24741307 IC50 = 15000 nM T19244 CQ35ZB 24743795 IC50 > 50000 nM T19244 C8RC9P 24744325 IC50 > 10000 nM T19244 C0L8QY 24744859 IC50 = 11000 nM T19244 CC4GB1 24748513 IC50 = 20000 nM T19244 CSG9V8 24749508 IC50 > 100000 nM T19244 C6JF2R 24753412 IC50 = 12000 nM T19244 C4CY3V 24753607 IC50 = 29000 nM T19244 CP1E4R 24753786 IC50 > 100000 nM T19244 COAY09 24753878 IC50 = 19000 nM T19244 C25HKJ 24758044 IC50 > 40000 nM T19244 CJL67N 24759089 IC50 > 10000 nM T19244 C3OY6A 24759171 IC50 = 3 nM T19244 CR9ZI2 24764491 IC50 > 50000 nM T19244 CG23NJ 24768399 IC50 = 10000 nM T19244 C3P7IS 24768572 IC50 = 36500 nM T19244 C85ELO 24771983 IC50 = 4400 nM T19244 C9EKA0 24778067 Ki = 101 nM T19244 C6ORA8 24783140 IC50 > 10000 nM T19244 CXSZ08 24783396 IC50 = 1700 nM T19244 CUM03S 24798754 IC50 > 50000 nM T19244 CR48VC 24809711 IC50 = 8000 nM T19244 CY8X0J 24811794 IC50 > 30000 nM T19244 C35JHQ 24812745 IC50 = 900 nM T19244 CK02ZF 24812771 IC50 > 50000 nM T19244 C6H2KZ 24817638 IC50 > 30000 nM T19244 CLP68C 24823665 IC50 = 7.8 nM T19244 CRV5C7 24823814 IC50 = 39 nM T19244 C73LOX 24824080 IC50 = 63 nM T19244 CF75DJ 24824494 IC50 = 9700 nM T19244 CUE62F 24824744 IC50 = 1000 nM T19244 C5Q3ZJ 24825257 IC50 = 200 nM T19244 CV1P6N 24825260 IC50 = 200 nM T19244 CUX47I 24825261 IC50 = 200 nM T19244 C7G6OT 24825262 IC50 = 1700 nM T19244 C1B8TF 24825267 IC50 = 6000 nM T19244 C06COB 24825268 IC50 = 13000 nM T19244 C47QTG 24825269 IC50 = 35000 nM T19244 CJ16YD 24825270 IC50 = 11000 nM T19244 CO1BL7 24825271 IC50 = 2500 nM T19244 CV0UB1 24825272 IC50 = 8700 nM T19244 CQN3Z7 24825710 IC50 = 25000 nM T19244 CZ5T2C 24825713 IC50 = 20000 nM T19244 CN4Z2J 24825807 IC50 = 200 nM T19244 C2MA5J 24825905 IC50 = 5000 nM T19244 C7ZQ1U 24826095 IC50 = 4000 nM T19244 CJ6Z9E 24826945 IC50 = 6000 nM T19244 CA29CU 24826946 IC50 = 1000 nM T19244 CY6QD7 24826947 IC50 = 4000 nM T19244 CM2Y0L 24827043 IC50 <= 1000 nM T19244 CLM16X 24827044 IC50 = 7000 nM T19244 C2IB1S 24827045 IC50 = 3000 nM T19244 CHS35U 24827139 IC50 = 1000 nM T19244 C6OJ5C 24827142 IC50 = 300 nM T19244 C2K1OE 24830571 IC50 = 12000 nM T19244 CR7X1M 24856034 IC50 = 8600 nM T19244 C61KPI 24856363 IC50 = 4400 nM T19244 CB4LY1 24857598 IC50 > 10000 nM T19244 CSR8J4 24857759 IC50 > 25000 nM T19244 CM8BS1 24879232 IC50 = 1320 nM T19244 CX79IO 24882359 IC50 > 20000 nM T19244 CKRF92 24888487 IC50 = 17000 nM T19244 CU1G7V 24888656 IC50 = 3700 nM T19244 CF2H0Z 24888658 IC50 = 13000 nM T19244 CH9JZ4 24888820 IC50 = 10000 nM T19244 C45AQE 24889168 IC50 = 4200 nM T19244 C0Z2TG 24889346 IC50 = 3400 nM T19244 CDQ9I1 24889676 IC50 = 4600 nM T19244 CY8I0R 24889679 IC50 = 8600 nM T19244 C6NVP1 24889840 IC50 = 19000 nM T19244 CTE1I8 24889844 IC50 = 3200 nM T19244 CU18OW 24890344 IC50 = 630 nM T19244 CUZ31Q 24890346 IC50 = 860 nM T19244 C32TKP 24890348 IC50 = 3200 nM T19244 CBK4Z3 24890525 IC50 = 17000 nM T19244 CU4HV5 24890872 IC50 = 2500 nM T19244 CNQ6I4 24894028 IC50 > 20000 nM T19244 CW3C5U 24896569 IC50 = 64 nM T19244 CDI7N3 24897002 IC50 > 50000 nM T19244 C8GN9W 24899993 IC50 > 50000 nM T19244 CZSA05 24899995 IC50 > 50000 nM T19244 CIZ6O1 24900235 IC50 > 50000 nM T19244 C61ARF 24900236 IC50 > 50000 nM T19244 C7J4ZQ 24900259 IC50 > 40000 nM T19244 CC4K1P 24949545 IC50 = 1000 nM T19244 C17QKF 24949548 IC50 = 2900 nM T19244 CCA9G2 24949700 IC50 = 1400 nM T19244 CFU0T1 24949702 IC50 = 500 nM T19244 CE79PI 24949704 IC50 = 15000 nM T19244 CI7NG8 24951587 IC50 > 8000 nM T19244 CLZ23U 24951610 IC50 > 30000 nM T19244 CNP3T1 24951733 IC50 > 50000 nM T19244 CEGV39 24951942 IC50 > 10000 nM T19244 C9EH3S 24951943 IC50 > 10000 nM T19244 CW9UN1 24951944 IC50 > 10000 nM T19244 CP98YL 24951946 IC50 > 10000 nM T19244 CJ43DG 24954671 IC50 = 200 nM T19244 C3VO7Q 24960588 IC50 = 14000 nM T19244 CZ89IP 24961687 IC50 = 4000 nM T19244 CW4X0E 24962988 IC50 > 3000 nM T19244 CB68JF 24963286 IC50 > 50000 nM T19244 CAN92Q 24968874 IC50 = 4100 nM T19244 CE95WV 24970356 IC50 = 150 nM T19244 CQ2Z7T 24985115 IC50 = 7000 nM T19244 CM7HQ5 24985395 IC50 > 20000 nM T19244 CEJ74C 24985745 IC50 > 20000 nM T19244 C27WVS 24986404 IC50 = 8000 nM T19244 C94AHE 24988956 IC50 = 10000 nM T19244 C14EFU 24990122 IC50 = 1200 nM T19244 C80LEK 24990485 IC50 = 2400 nM T19244 CMD98H 24990837 IC50 = 11000 nM T19244 CNMD47 24990839 IC50 = 7900 nM T19244 C0I5NG 24991884 IC50 = 18000 nM T19244 CL83OS 24992519 IC50 > 30000 nM T19244 CK0NZ8 24993163 IC50 = 1000 nM T19244 C8KIP6 24993178 IC50 > 30000 nM T19244 CD8U2B 24993500 IC50 > 30000 nM T19244 CCDF20 24994127 IC50 > 30000 nM T19244 CDF57P 24995525 IC50 = 1258.93 nM T19244 CJM8R0 24996322 IC50 > 30000 nM T19244 CZ6T5Q 25009937 IC50 > 29000 nM T19244 CU7G9E 25010550 IC50 < 10000 nM T19244 C32AUW 25013308 IC50 > 10000 nM T19244 C4E9IK 25015611 IC50 = 9000 nM T19244 CCE8S3 25015613 IC50 = 7000 nM T19244 CP13LW 25016311 IC50 = 3000 nM T19244 C91QFN 25019282 IC50 = 47000 nM T19244 CMU30E 25022640 IC50 > 100000 nM T19244 CF67EB 25023856 IC50 = 10000 nM T19244 C0L9PQ 25023857 IC50 < 10000 nM T19244 CA2T1X 25023858 IC50 < 10000 nM T19244 C7SKU1 25023859 IC50 < 10000 nM T19244 CA20NZ 25025581 IC50 > 9000 nM T19244 CPJD86 25025779 IC50 > 4000 nM T19244 CDX2C6 25025977 IC50 > 8000 nM T19244 C0LO9C 25028373 IC50 = 13000 nM T19244 CKLQ76 25028375 IC50 = 3000 nM T19244 CDKJ78 25033361 IC50 > 40000 nM T19244 CXDF80 25034348 IC50 > 200000 nM T19244 CR3I9Y 25050394 EC50 = 55000 nM T19244 CVQS96 25052767 IC50 > 25000 nM T19244 CZO27W 25054032 IC50 > 30000 nM T19244 C7EQ5T 25054288 IC50 > 10000 nM T19244 CN2G3K 25054307 IC50 > 30000 nM T19244 C7EXD5 25054568 IC50 > 30000 nM T19244 C1PKF0 25056080 IC50 > 10000 nM T19244 CFHO90 25056112 IC50 > 30000 nM T19244 C6Z3CE 25057124 IC50 > 10000 nM T19244 CH6AU8 25057408 IC50 > 30000 nM T19244 C0B7RT 25057409 IC50 > 30000 nM T19244 C3AT0H 25057667 IC50 > 30000 nM T19244 CH7YC4 25057933 IC50 > 30000 nM T19244 CGMN97 25067404 IC50 > 30000 nM T19244 CMJ1F7 25067546 IC50 > 50000 nM T19244 CMH41V 25069448 IC50 = 270 nM T19244 CBY3O2 25070582 IC50 > 30000 nM T19244 CBRM65 25074167 IC50 = 1250 nM T19244 C1AGW7 25093241 IC50 = 8400 nM T19244 CH90KV 25097876 IC50 > 10000 nM T19244 CAO38V 25098429 IC50 > 10000 nM T19244 CF7ON5 25099235 IC50 > 50000 nM T19244 CUYI02 25101821 IC50 > 10000 nM T19244 C0K9HA 25110600 IC50 > 14000 nM T19244 CNW3T2 25113689 Ki = 4.2 nM T19244 C8BZ0T 25117985 IC50 = 2400 nM T19244 CK06LQ 25118337 IC50 = 7300 nM T19244 CQE1C2 25118338 IC50 > 10000 nM T19244 CKRN07 25118654 IC50 > 50000 nM T19244 CZ96TL 25118804 IC50 > 50000 nM T19244 C8T7NC 25118805 IC50 > 50000 nM T19244 CM7WO3 25122581 IC50 = 2000 nM T19244 CDO26T 25129042 IC50 > 31622.78 nM T19244 COD4T6 25138286 IC50 = 1000 nM T19244 C9Z6UG 25138295 IC50 > 100000 nM T19244 CHS25Z 25141776 IC50 > 5000 nM T19244 CE93TF 25141777 IC50 > 5000 nM T19244 C1AIH7 25141896 IC50 > 5000 nM T19244 CWF5Z3 25143506 IC50 > 30000 nM T19244 CFS3N9 25144422 IC50 > 20000 nM T19244 C78YWA 25145716 IC50 > 20000 nM T19244 C8AC0Y 25154864 IC50 > 5000 nM T19244 CGH08V 25164128 IC50 = 31000 nM T19244 C3NVW5 25165471 IC50 = 8000 nM T19244 CF9KY4 25165474 IC50 > 8000 nM T19244 CH06WV 25168930 IC50 > 10000 nM T19244 C5TJD2 25172265 IC50 > 10000 nM T19244 CJMZ37 25174150 IC50 = 340 nM T19244 CFA08V 25179508 Ki = 9740 nM T19244 CH4YU2 25179509 Ki = 3670 nM T19244 CHOA95 25179510 Ki = 24080 nM T19244 CKJ80S 25179511 Ki = 76190 nM T19244 C1C2WL 25179512 Ki = 33 nM T19244 CBI3Q5 25179706 Ki = 10670 nM T19244 C4L1JK 25179707 Ki = 113 nM T19244 C64PZD 25179708 Ki = 152 nM T19244 C8R2DK 25179709 Ki > 43500 nM T19244 CAU8R2 25179901 Ki = 11 nM T19244 CURI31 25179902 Ki = 8550 nM T19244 CXD47A 25179903 Ki > 20600 nM T19244 CEU4D0 25179904 Ki = 12 nM T19244 CN78BM 25179905 Ki = 1890 nM T19244 C9K1CW 25179906 Ki = 9 nM T19244 CUQ7D1 25180096 Ki > 37850 nM T19244 CH04GE 25180097 Ki = 1250 nM T19244 CXV3O9 25180098 Ki = 1320 nM T19244 C0XHA2 25180109 IC50 = 125000 nM T19244 C90UKD 25180304 IC50 = 16300 nM T19244 C6ZE9H 25180500 IC50 = 12900 nM T19244 CK6Z9J 25181419 IC50 = 17000 nM T19244 C6EWF1 25183622 IC50 > 30000 nM T19244 C5C7GH 25184832 IC50 > 10000 nM T19244 CSU0B5 25189891 IC50 > 15000 nM T19244 C04QGB 25190493 IC50 > 89000 nM T19244 CV3TA6 25192021 IC50 > 12500 nM T19244 C9UL8Y 25192468 IC50 = 7600 nM T19244 C7A8UE 25192471 IC50 > 25000 nM T19244 CH3L6V 25192656 IC50 > 10000 nM T19244 CDC4S5 25195002 IC50 = 9200 nM T19244 C8CY6O 25205318 IC50 > 10000000 nM T19244 CY1M9Q 25205319 IC50 > 10000000 nM T19244 CLFM35 25206064 IC50 = 5100 nM T19244 CSGI69 25207352 IC50 = 12000 nM T19244 C37YTG 25210603 IC50 > 10000 nM T19244 CTQM87 25210756 IC50 > 25000 nM T19244 CE7BA0 25210873 IC50 > 10000 nM T19244 C2UQJ6 25211598 EC50 = 29000 nM T19244 CKI86X 25211805 EC50 > 60000 nM T19244 CHW2X0 25211910 EC50 > 60000 nM T19244 CXH7F8 25218692 IC50 > 20000 nM T19244 CUN19O 25218744 IC50 = 7000 nM T19244 CJ65AE 25226377 IC50 > 50000 nM T19244 CW9JM2 25256832 IC50 > 10000 nM T19244 C3GC7P 25256833 IC50 > 10000 nM T19244 C4N8BX 25261287 IC50 = 1800 nM T19244 CWYJ73 25261449 IC50 = 17000 nM T19244 CU1Y6R 25261451 IC50 = 16000 nM T19244 CL2NO1 25261454 IC50 > 25000 nM T19244 C1IW5M 25261456 IC50 > 33000 nM T19244 CRJ8H4 25261457 IC50 > 25000 nM T19244 CV5FB3 25261927 IC50 = 25000 nM T19244 C5E3ZH 25265089 IC50 > 100000 nM T19244 CJ32HC 25265835 IC50 = 4000 nM T19244 CGQ8D3 25270849 IC50 = 8400 nM T19244 CI1G2C 26873419 IC50 = 18900 nM T19244 CC9S5U 28412206 IC50 < 100 nM T19244 C0FA2X 40680501 IC50 = 39900 nM T19244 CE63OB 40700807 IC50 > 20000 nM T19244 CHW3D1 40700815 IC50 > 20000 nM T19244 CBH1P0 42210730 IC50 > 30000 nM T19244 CT0NF6 42415086 IC50 > 30000 nM T19244 CA25BL 42603033 IC50 = 82000 nM T19244 CKH3P1 42606928 IC50 > 40000 nM T19244 C1YO7H 42618040 EC50 = 33000 nM T19244 C0I4MK 42618066 EC50 = 22000 nM T19244 CGU3N8 42618068 EC50 = 25000 nM T19244 CY4LG8 42622934 IC50 > 75000 nM T19244 C73LBP 42625213 IC50 = 4400 nM T19244 C2H6QR 42625218 IC50 = 2000 nM T19244 CJPW47 42625379 IC50 = 990 nM T19244 CW7A0V 42625382 IC50 = 4700 nM T19244 CT0H2G 42625474 IC50 = 12000 nM T19244 CGI02C 42625475 IC50 = 1500 nM T19244 CS34QO 42625476 IC50 = 19000 nM T19244 CJ8LY0 42626024 IC50 = 6000 nM T19244 CS04KE 42629368 IC50 > 20000 nM T19244 CYGN52 42629369 IC50 > 20000 nM T19244 C4P1IM 42643589 IC50 > 10000 nM T19244 CX9SM6 42643591 IC50 < 10000 nM T19244 C96FIN 42644084 IC50 > 10000 nM T19244 C8BI5F 42644088 IC50 > 10000 nM T19244 CREJ31 42646199 IC50 > 10000 nM T19244 CKZ76R 42646202 IC50 < 10000 nM T19244 C81NVM 42646450 IC50 < 10000 nM T19244 CVBO78 42647178 IC50 > 10000 nM T19244 CZF5G9 42916879 IC50 = 3000 nM T19244 C5E6UL 43388611 IC50 = 50000 nM T19244 CS40ML 44123747 IC50 > 50000 nM T19244 CS0H1B 44125704 IC50 > 50000 nM T19244 C7VOU1 44126023 IC50 = 800 nM T19244 C47OXT 44128987 IC50 > 50000 nM T19244 CN5O1Y 44129065 IC50 = 27000 nM T19244 CX7W2E 44132009 IC50 = 42000 nM T19244 CXS43I 44132271 IC50 > 25000 nM T19244 CA7HI4 44137226 IC50 = 7300 nM T19244 CMJI64 44137938 IC50 = 1200 nM T19244 CG73ST 44138103 IC50 > 30000 nM T19244 C6QY9W 44143257 IC50 = 60000 nM T19244 C5G4LN 44159411 IC50 > 30000 nM T19244 CHI65U 44159530 IC50 = 18000 nM T19244 CMNH53 44159772 IC50 = 18000 nM T19244 C38DTW 44160263 IC50 > 40000 nM T19244 CO9AY2 44182947 IC50 > 25000 nM T19244 CPF50A 44184875 IC50 > 24000 nM T19244 CBPV86 44188851 IC50 = 1000 nM T19244 CWM71O 44188852 IC50 > 25000 nM T19244 C2XE7Y 44189733 IC50 > 100000 nM T19244 C5AK1N 44190592 IC50 = 5600 nM T19244 CSN2I3 44190675 IC50 = 10000 nM T19244 C6SG0O 44192200 IC50 = 358000 nM T19244 C5L6WO 44194849 IC50 > 10000 nM T19244 CRU6J3 44205381 IC50 = 16000 nM T19244 CZ29JY 44205724 IC50 > 30000 nM T19244 C5RL9M 44215838 IC50 > 20000 nM T19244 C7VWX5 44220300 IC50 > 10000 nM T19244 C2O0NL 44230575 IC50 > 20000 nM T19244 CX4YL8 44232522 IC50 > 10000 nM T19244 CQ13MH 44234032 IC50 > 50000 nM T19244 C7UY5F 44235863 IC50 > 10000 nM T19244 CX2W8Y 44236320 IC50 > 10000 nM T19244 C8LN0U 44236321 IC50 < 10000 nM T19244 CK4S5Y 44236322 IC50 < 10000 nM T19244 C4W0SH 44247585 IC50 > 40000 nM T19244 CDOA12 44249906 IC50 > 41000 nM T19244 C8P2LE 44250288 IC50 > 10000 nM T19244 CLY1A3 44251218 IC50 = 10000 nM T19244 C8BXD9 44251608 IC50 > 10000 nM T19244 CNO97U 44255810 IC50 > 20000 nM T19244 CV7J8H 44265173 IC50 = 2000 nM T19244 CTR62D 44265213 IC50 = 3000 nM T19244 C6HO3T 44335329 IC50 = 7400 nM T19244 C7S2ZI 44340870 IC50 = 8590 nM T19244 CE13FX 44341241 IC50 = 40000 nM T19244 CX65PH 44341461 IC50 = 32800 nM T19244 C0KD4U 44346053 IC50 > 2000 nM T19244 CH0O5Q 44346322 IC50 > 2000 nM T19244 C6QM2Z 44346781 IC50 = 20000 nM T19244 C5OQ2K 44366980 IC50 = 19200 nM T19244 CKF5G6 44367711 IC50 = 24000 nM T19244 CW48BI 44367781 IC50 = 30000 nM T19244 C6C8QK 44382913 Ki = 16000 nM T19244 C7F3SW 44383264 Ki = 13600 nM T19244 CM6V4C 44388606 IC50 = 79500 nM T19244 CKV1H9 44388612 IC50 > 300000 nM T19244 CGU79D 44388657 IC50 = 208000 nM T19244 C4X2OS 44396541 IC50 > 50000 nM T19244 CY80RP 44396542 IC50 = 480 nM T19244 C9P7QL 44399862 IC50 = 50 nM T19244 C4NUA0 44402523 IC50 > 30000 nM T19244 C3X6LO 44403285 IC50 = 19490 nM T19244 CKZX07 44403288 IC50 > 100000 nM T19244 CUGE51 44403300 IC50 = 3900 nM T19244 CAN69Y 44409279 IC50 < 50 nM T19244 C0SXD3 44410799 IC50 > 5000 nM T19244 CR4HX5 44410840 IC50 > 5000 nM T19244 C73OZJ 44410841 IC50 > 5000 nM T19244 CYCU18 44410874 IC50 = 6800 nM T19244 CY2F3Q 44420235 IC50 > 10000 nM T19244 CH1R7M 44420600 IC50 > 10000 nM T19244 CU52GB 44425701 IC50 = 47000 nM T19244 CX8TR0 44425719 IC50 = 17000 nM T19244 C40HMY 44427622 IC50 > 40000 nM T19244 CYM7Q6 44427624 IC50 > 40000 nM T19244 CV7LZ9 44427625 IC50 > 40000 nM T19244 CTO57H 44427626 IC50 > 40000 nM T19244 C9PLA8 44427627 IC50 > 40000 nM T19244 CAWL05 44428924 IC50 > 10000 nM T19244 CZ4W6P 44430775 IC50 = 9000 nM T19244 CTB82G 44431744 IC50 > 50000 nM T19244 CL6B7S 44431775 IC50 = 15000 nM T19244 C9LM7U 44433789 IC50 = 26000 nM T19244 CWDJ93 44433797 IC50 = 69000 nM T19244 CU67NA 44433798 IC50 > 100000 nM T19244 CNU4B6 44433799 IC50 = 43000 nM T19244 C5V7WE 44433800 IC50 = 47000 nM T19244 CBP25Q 44433802 IC50 = 89000 nM T19244 CB1SD9 44433803 IC50 = 9000 nM T19244 CT7Q2I 44440397 IC50 = 66 nM T19244 CP2G6L 44440493 IC50 = 1400 nM T19244 CXSQ75 44440525 IC50 = 17600 nM T19244 C2VAG9 44440645 IC50 > 10000 nM T19244 C08ZST 44440659 IC50 > 10000 nM T19244 CR3PM7 44440662 IC50 > 10000 nM T19244 CCSI57 44440665 IC50 > 10000 nM T19244 CT0C4I 44443093 IC50 > 20000 nM T19244 C8E1AC 44443094 IC50 = 14000 nM T19244 CZ6BK9 44443095 IC50 = 18000 nM T19244 CV5T2C 44443096 IC50 = 12000 nM T19244 CF1V8O 44443098 IC50 = 7000 nM T19244 CHZ48Q 44443101 IC50 = 4000 nM T19244 CQ53TV 44443130 IC50 > 19000 nM T19244 CEZ6U8 44443131 IC50 > 16000 nM T19244 CN4XZ6 44443132 IC50 > 9000 nM T19244 CV5CK0 44443532 IC50 = 1470 nM T19244 C5HMU1 44446711 IC50 = 1500 nM T19244 CXPD58 44453913 IC50 = 3000 nM T19244 C9YUM3 44453941 IC50 = 670 nM T19244 CPM4W2 44454303 IC50 > 66000 nM T19244 CZ39GO 44455035 IC50 > 10000 nM T19244 CWL42H 44457199 IC50 = 2700 nM T19244 C2KMI6 44469322 IC50 = 1720 nM T19244 C1ZBJ3 44469819 IC50 > 6000 nM T19244 C2QK4J 44472590 IC50 > 100000 nM T19244 CQ8C3F 44472591 IC50 > 100000 nM T19244 CWN95E 44472610 IC50 > 100000 nM T19244 C1H2ZT 44472612 IC50 > 100000 nM T19244 CC75ON 44473086 IC50 = 10000 nM T19244 CUZ97H 44473093 IC50 = 122000 nM T19244 CSFM32 44473094 IC50 = 10000 nM T19244 C2OT5K 44473095 IC50 = 9000 nM T19244 C4H0DY 44473096 IC50 = 12000 nM T19244 C7S8OZ 44473097 IC50 = 122000 nM T19244 CO19AD 44473098 IC50 = 22000 nM T19244 CTP32R 44473099 IC50 = 24000 nM T19244 CM37YN 44475195 IC50 = 10 nM T19244 CSBL94 44475353 IC50 > 10 nM T19244 C2ZI9A 44475365 IC50 = 2000 nM T19244 CSB0C1 44475367 IC50 = 7000 nM T19244 C3GYC0 44475943 IC50 >= 100000 nM T19244 CX9TJ4 44476890 IC50 = 43000 nM T19244 C7TK5E 44479928 IC50 = 1995.26 nM T19244 CB1I8L 44479933 IC50 > 100000 nM T19244 CEF20J 44479934 IC50 = 63095.73 nM T19244 C0RYL8 44480178 IC50 = 15848.93 nM T19244 C42CKX 44480181 IC50 = 12589.25 nM T19244 CQE20D 44480441 IC50 = 39810.72 nM T19244 C78ALJ 44480442 IC50 = 39810.72 nM T19244 C2XW9P 44480443 IC50 = 39810.72 nM T19244 CT38MK 44480444 IC50 = 31622.78 nM T19244 CUA9F0 44512094 IC50 > 50000 nM T19244 C4M9FH 44512619 IC50 > 40000 nM T19244 CU80BP 44517743 IC50 > 21000 nM T19244 CS9H0L 44517795 IC50 > 50000 nM T19244 CKI82C 44518336 IC50 > 1000 nM T19244 CSO35V 44520546 IC50 = 251.19 nM T19244 CJCB39 44520861 IC50 = 13000 nM T19244 CJA36X 44533150 IC50 = 2000 nM T19244 C9N1BU 44539192 IC50 > 20000 nM T19244 C14SNF 44539764 IC50 > 30000 nM T19244 CLMY52 44539967 IC50 > 10000 nM T19244 CMW56J 44539973 IC50 > 30000 nM T19244 C0RA9E 44540072 IC50 > 30000 nM T19244 C27TZY 44543970 IC50 = 12000 nM T19244 CK1Z8P 44545482 IC50 = 12000 nM T19244 CECD12 44547033 IC50 = 21400 nM T19244 CX13MK 44547414 IC50 = 34800 nM T19244 CP6R2X 44551848 IC50 = 13000 nM T19244 C4RB7W 44555352 IC50 > 10000 nM T19244 C5EX1K 44555473 IC50 > 10000 nM T19244 CV1IL5 44565796 IC50 > 10000 nM T19244 CQ12FA 44567235 Ki = 41 nM T19244 C9MAV5 44567236 Ki = 23 nM T19244 C8XC6Y 44567391 Ki = 4870 nM T19244 C6MVD1 44567392 Ki = 6740 nM T19244 C69RCJ 44567393 Ki = 1420 nM T19244 CR9PB8 44567394 Ki = 656 nM T19244 C7AI9D 44567410 Ki = 6480 nM T19244 CY7B0L 44567411 Ki = 3120 nM T19244 CS7G2D 44567412 Ki = 44.34 nM T19244 CB5S9R 44569927 IC50 = 40000 nM T19244 C6Q5DK 44569945 IC50 = 800 nM T19244 CBET53 44570224 IC50 = 10000 nM T19244 CP32DL 44570256 IC50 = 27000 nM T19244 CVO8L1 44570275 IC50 = 4000 nM T19244 CP0F6X 44571381 IC50 = 610 nM T19244 CS3A6G 44571481 IC50 = 650 nM T19244 CAJM40 44571482 IC50 = 180 nM T19244 CI9PS7 44571483 IC50 = 210 nM T19244 CK1BM3 44571524 IC50 = 2400 nM T19244 C5L7FR 44571525 IC50 = 9400 nM T19244 CV6DF8 44571636 IC50 > 33000 nM T19244 C1P8RS 44571637 IC50 > 33000 nM T19244 C8VRB1 44571638 IC50 > 33000 nM T19244 C7WNI0 44571639 IC50 > 33000 nM T19244 C6AB7R 44571788 IC50 = 12000 nM T19244 C2VSW5 44571789 IC50 = 2300 nM T19244 CZ39EI 44571790 IC50 = 1940 nM T19244 C2OD8E 44571903 IC50 = 450 nM T19244 CIBP35 44571952 IC50 = 32000 nM T19244 CWP80I 44571963 IC50 = 9800 nM T19244 CCM0D8 44571965 IC50 = 4900 nM T19244 CO3L8Z 44571998 IC50 = 14000 nM T19244 CCY14Q 44571999 IC50 = 2100 nM T19244 C67KIU 44572000 IC50 = 7230 nM T19244 CLG7X2 44572011 IC50 = 1800 nM T19244 CPB6A7 44572040 IC50 = 1900 nM T19244 C1XW9C 44572041 IC50 = 680 nM T19244 CYLI30 44572042 IC50 = 50 nM T19244 C9IPZ6 44572058 IC50 = 400 nM T19244 CZ56HX 44574108 IC50 > 5000 nM T19244 CFJB16 44578266 IC50 > 3000 nM T19244 CG80OC 44578914 IC50 > 50000 nM T19244 C7LAT0 44578954 IC50 > 50000 nM T19244 CBG04P 44578955 IC50 > 50000 nM T19244 CA3FO8 44578956 IC50 = 14700 nM T19244 CA16QJ 44578957 IC50 > 50000 nM T19244 CFH01N 44578958 IC50 > 50000 nM T19244 CMA26F 44578959 IC50 > 50000 nM T19244 C79PYS 44578960 IC50 > 50000 nM T19244 CF39ON 44578961 IC50 > 50000 nM T19244 C4KI0B 44579189 IC50 > 50000 nM T19244 C1I0QG 44579190 IC50 > 50000 nM T19244 C6VFZ3 44579191 IC50 > 50000 nM T19244 C1O5ET 44579232 IC50 > 50000 nM T19244 CY8NJ4 44579233 IC50 > 50000 nM T19244 CSLC36 44579234 IC50 > 50000 nM T19244 CBK23W 44579235 IC50 > 50000 nM T19244 CS2KV6 44579236 IC50 > 50000 nM T19244 C60CAD 44579237 IC50 > 50000 nM T19244 CX85MD 44579273 IC50 > 50000 nM T19244 C0IP7C 44583234 IC50 < 10000 nM T19244 C6HTC1 44583235 IC50 > 10000 nM T19244 CZJU04 44583236 IC50 < 10000 nM T19244 C3TYW0 44583237 IC50 < 10000 nM T19244 CCL9R0 44583238 IC50 < 10000 nM T19244 COX7F1 44583287 IC50 < 10000 nM T19244 CFT74N 44583289 IC50 > 10000 nM T19244 CC19TZ 44583290 IC50 > 10000 nM T19244 C90RAV 44583349 IC50 > 10000 nM T19244 CK81NJ 44583350 IC50 = 10000 nM T19244 C20VTN 44583351 IC50 > 10000 nM T19244 CD5U3A 44583352 IC50 < 10000 nM T19244 C9G7VT 44583353 IC50 > 10000 nM T19244 C6QF4O 44583354 IC50 = 7600 nM T19244 C48AQR 44583355 IC50 = 10000 nM T19244 CG5X0M 44583356 IC50 < 10000 nM T19244 CUG9Y0 44583357 IC50 > 10000 nM T19244 CRE9Q2 44583561 IC50 = 14000 nM T19244 C9AP1O 44583590 IC50 = 5800 nM T19244 CO6XB8 44583591 IC50 = 6500 nM T19244 CM6Y4F 44583614 IC50 = 4700 nM T19244 CR13XJ 44583631 IC50 = 2900 nM T19244 C53KBN 44583632 IC50 = 1100 nM T19244 CK27DJ 44583633 IC50 = 5600 nM T19244 C9EX2M 44583647 IC50 = 23000 nM T19244 C7K6YM 44583648 IC50 = 2500 nM T19244 CZ2D3P 44583663 IC50 = 97000 nM T19244 C5XD4S 44583664 IC50 = 5300 nM T19244 CKW9Y5 44583665 IC50 = 5600 nM T19244 CDZN40 44583666 IC50 = 14000 nM T19244 C0IFL7 44583667 IC50 = 21000 nM T19244 CHR03D 44583679 IC50 = 4200 nM T19244 CHG2M3 44586212 IC50 > 100000 nM T19244 CCS62T 44587583 IC50 = 316.23 nM T19244 C9RA0C 44589548 EC50 = 10000 nM T19244 CWKP93 44589698 IC50 = 5000 nM T19244 CS4JP5 44589733 IC50 = 1800 nM T19244 CEPG12 44589734 IC50 = 17000 nM T19244 CZVO54 44589735 IC50 = 3000 nM T19244 CPB1G7 44589736 IC50 = 5000 nM T19244 CH54CO 44589824 IC50 = 2320 nM T19244 C89LHN 44589825 IC50 = 2270 nM T19244 C70MSI 44593549 IC50 = 23000 nM T19244 CCA7K5 44593648 IC50 > 50000 nM T19244 C64ZKC 44593664 IC50 > 10000 nM T19244 C01BFQ 44593665 IC50 > 10000 nM T19244 CE97GB 44596160 IC50 > 20000 nM T19244 C4ID9A 44602971 IC50 > 30000 nM T19244 C7I4EY 44603096 IC50 > 30000 nM T19244 C4MOE2 44603271 IC50 = 1300 nM T19244 C89VRG 44605616 IC50 > 10000 nM T19244 CZD25I 44605617 IC50 > 10000 nM T19244 CXQ19C 44610104 IC50 = 6000 nM T19244 C0WVZ1 44622338 IC50 > 30000 nM T19244 CL26YD 44622339 IC50 > 30000 nM T19244 CA7EQ2 44622340 IC50 > 30000 nM T19244 C23ORN 44622341 IC50 > 30000 nM T19244 C2JIX6 44622342 IC50 > 30000 nM T19244 CNI29G 44622416 IC50 > 30000 nM T19244 C9KUD5 44622417 IC50 > 30000 nM T19244 C4Q7JB 44622418 IC50 > 30000 nM T19244 C12SGH 44622499 IC50 > 30000 nM T19244 C2OUJ0 44624151 IC50 > 5000 nM T19244 C0N6DO 44625908 IC50 = 8000 nM T19244 CXD90A 44625911 IC50 = 20100 nM T19244 C85ZIF 44626928 IC50 > 10000 nM T19244 C4BYG5 44626929 IC50 > 10000 nM T19244 CQE59L 44627133 IC50 > 10000 nM T19244 CDQ47G 44629236 IC50 > 25000 nM T19244 CH3SF9 44631836 IC50 > 27000 nM T19244 CPG61Y 44718445 IC50 > 20000 nM T19244 C3Q7BW 44816514 IC50 > 30000 nM T19244 C85DWU 44816692 IC50 = 4000 nM T19244 CJ0F5Q 44819015 IC50 = 16000 nM T19244 CN21OS 44819193 IC50 > 30000 nM T19244 CQI0D4 45102707 IC50 = 400 nM T19244 CSEP-69 45102708 IC50 = 200 nM T19244 CGCZ64 45102767 IC50 > 50000 nM T19244 C7NFZ1 45110765 IC50 = 8700 nM T19244 CR6UW4 45112038 IC50 > 50000 nM T19244 CUL67Y 45202552 IC50 > 30000 nM T19244 C4KRT0 45254002 IC50 = 1200 nM T19244 C1K0ZH 45259193 IC50 > 10000 nM T19244 CB9QZ6 45263405 IC50 = 23000 nM T19244 CQ85WF 45263621 IC50 > 10000 nM T19244 CUT2B4 45267348 IC50 > 10000 nM T19244 C53DIE 45267853 IC50 = 14000 nM T19244 CJH3A2 45268206 IC50 > 10000 nM T19244 CULJ91 45268456 IC50 = 10000 nM T19244 C4WR0V 45269087 IC50 > 10000 nM T19244 CRPS25 45269096 IC50 > 10000 nM T19244 C7BNY6 45269104 IC50 = 10000 nM T19244 CB5O6V 45269307 IC50 = 18000 nM T19244 CS1Q2X 45269947 IC50 > 10000 nM T19244 C1BE5U 45269948 IC50 > 10000 nM T19244 CG1H9N 45269950 IC50 < 10000 nM T19244 C03ETI 45270148 IC50 > 30000 nM T19244 C1NT2M 45270771 IC50 > 10000 nM T19244 CA05IG 45270778 IC50 > 10000 nM T19244 CZ7MK9 45270788 IC50 < 10000 nM T19244 CY70SI 45270983 IC50 > 30000 nM T19244 C2XH3A 45270987 IC50 > 30000 nM T19244 C9TM2P 45271593 IC50 > 10000 nM T19244 C06YAD 45271599 IC50 > 10000 nM T19244 CG0I8P 45271610 IC50 < 10000 nM T19244 C6FBH0 45271618 IC50 > 10000 nM T19244 C71VIG 45272510 IC50 > 10000 nM T19244 C05EDY 45272511 IC50 > 10000 nM T19244 C35DUQ 45272700 IC50 = 17000 nM T19244 CKUI32 45272704 IC50 = 15000 nM T19244 CD62AH 45273373 IC50 > 10000 nM T19244 CMN39U 45273380 IC50 > 10000 nM T19244 C3U7KT 45273637 IC50 > 30000 nM T19244 CZ71RN 45278805 IC50 = 9700 nM T19244 CYOW10 45377016 IC50 = 17390 nM T19244 C7D3LB 45377018 IC50 = 17253 nM T19244 C25PTU 45377580 IC50 = 1347 nM T19244 C8ELI4 45378010 IC50 = 2286 nM T19244 CMU6Z8 45379828 IC50 > 6000 nM T19244 CNQT48 45379947 IC50 > 10000 nM T19244 C0CHF4 45482789 IC50 > 10000 nM T19244 CX90YO 45484534 IC50 = 1500 nM T19244 CZUI01 45484860 IC50 = 3300 nM T19244 C65ONH 45484861 IC50 > 5000 nM T19244 C6KC8V 45484873 IC50 > 5000 nM T19244 CVR40A 45484874 IC50 > 5000 nM T19244 CV78NM 45484881 IC50 > 5000 nM T19244 C5DEA7 45484892 IC50 = 4000 nM T19244 CXYK82 45484893 IC50 = 2200 nM T19244 CR8VF3 45484894 IC50 > 5000 nM T19244 C7TQ3Z 45484899 IC50 = 3400 nM T19244 CD7N4J 45484900 IC50 > 5000 nM T19244 CQ84RV 45484907 IC50 > 5000 nM T19244 C1K0IO 45484913 IC50 = 3700 nM T19244 C2J4VM 45484915 IC50 > 5000 nM T19244 CE6J7S 45484916 IC50 > 5000 nM T19244 CI4SP9 45484917 IC50 > 5000 nM T19244 CYA6U2 45484918 IC50 > 5000 nM T19244 CYWT18 45484919 IC50 > 5000 nM T19244 C1FZ3N 45484922 IC50 > 5000 nM T19244 CXD74W 45484923 IC50 > 5000 nM T19244 CDP3X6 45484930 IC50 > 5000 nM T19244 CQ90DC 45484931 IC50 > 5000 nM T19244 CQ3I9D 45484949 IC50 = 4200 nM T19244 CZU29D 45484950 IC50 = 3900 nM T19244 CW6M7Q 45484961 IC50 > 5000 nM T19244 C4TI0X 45484966 IC50 > 5000 nM T19244 CWNH93 45484967 IC50 > 5000 nM T19244 C5R0YZ 45484968 IC50 > 5000 nM T19244 C9E4UO 45484969 IC50 > 5000 nM T19244 CL32NJ 45488686 IC50 > 10000 nM T19244 C7UAT9 46174270 IC50 > 30000 nM T19244 CP12AF 46179404 IC50 = 1510 nM T19244 CS8TU3 46179405 IC50 = 7350 nM T19244 C2L5UH 46182745 IC50 = 8200 nM T19244 CPU02J 46190696 IC50 = 2187 nM T19244 CYAI40 46198106 IC50 = 3400 nM T19244 CTI0F8 46198107 IC50 = 3700 nM T19244 CJ9OY8 46198108 IC50 = 7100 nM T19244 CI9QH8 46198109 IC50 = 3700 nM T19244 CU3VQ1 46198110 IC50 = 500 nM T19244 C2P9ST 46198216 IC50 = 8600 nM T19244 CSEL57 46198325 IC50 = 21000 nM T19244 C2VIF3 46198326 IC50 = 2800 nM T19244 C6JWH5 46198327 IC50 = 3500 nM T19244 C13RUW 46198329 IC50 = 4400 nM T19244 CFYP54 46203897 IC50 = 32000 nM T19244 C21ICG 46212134 IC50 = 21400 nM T19244 C62GRO 46212391 IC50 = 5620 nM T19244 CN3BE0 46212588 IC50 = 6400 nM T19244 CC9X1M 46213938 IC50 > 30000 nM T19244 CPF0J9 46214673 IC50 > 30000 nM T19244 CAX31B 46216689 IC50 > 15000 nM T19244 C5AY6M 46220498 IC50 > 10000 nM T19244 CFS6Q5 46224644 IC50 = 330 nM T19244 CURS28 46224649 IC50 = 280 nM T19244 C75QAG 46224653 IC50 = 110 nM T19244 CB5HP0 46224657 IC50 = 350 nM T19244 CI3OC4 46224664 IC50 = 160 nM T19244 CS9D6X 46224668 IC50 = 1400 nM T19244 C5N2WP 46224669 IC50 = 4000 nM T19244 C6XQF5 46224670 IC50 = 1200 nM T19244 C72ZGS 46224672 IC50 = 2400 nM T19244 CNG16S 46224673 IC50 = 14000 nM T19244 CS0Y7O 46224677 IC50 = 1500 nM T19244 CJP6A9 46224678 IC50 = 2900 nM T19244 CR9J1L 46224680 IC50 = 680 nM T19244 CZS7L4 46224681 IC50 = 690 nM T19244 CJZL72 46224683 IC50 = 1500 nM T19244 CKQF01 46224685 IC50 = 1100 nM T19244 C15RNW 46224687 IC50 = 720 nM T19244 C81YIZ 46224688 IC50 = 2900 nM T19244 CRSM47 46224691 IC50 = 1300 nM T19244 C0RJG8 46224692 IC50 = 1100 nM T19244 CQC6J0 46224693 IC50 = 440 nM T19244 C2A5QX 46224699 IC50 = 1100 nM T19244 CPHQ30 46224702 IC50 = 1800 nM T19244 C7JXG3 46224705 IC50 = 160 nM T19244 CMYU19 46224706 IC50 = 3000 nM T19244 CHCT54 46226167 IC50 = 2000 nM T19244 CJ7T4D 46226168 IC50 = 2000 nM T19244 CGR9I8 46226169 IC50 = 2000 nM T19244 C6KER3 46226224 IC50 = 1000 nM T19244 CAH58K 46226225 IC50 = 1000 nM T19244 C53ODR 46226226 IC50 = 1000 nM T19244 CLG0E3 46226227 IC50 = 13000 nM T19244 C0W9DL 46226238 IC50 = 23000 nM T19244 CNG98O 46226239 IC50 = 300 nM T19244 CP8U5O 46226240 IC50 = 12000 nM T19244 C8NIK4 46226256 IC50 = 15000 nM T19244 CIL85Q 46226257 IC50 = 1000 nM T19244 CRJ5F7 46226258 IC50 = 1000 nM T19244 CCQ19F 46226276 IC50 = 1000 nM T19244 CAK5M4 46226277 IC50 = 30000 nM T19244 CQ6L5E 46226278 IC50 = 30000 nM T19244 CVJU38 46233842 IC50 = 13700 nM T19244 CQ9A7L 46234188 IC50 > 30000 nM T19244 C94GCA 46234349 IC50 > 30000 nM T19244 C8PZU1 46235580 IC50 = 4.5 nM T19244 C7OB2G 46235733 IC50 = 4010 nM T19244 CIGB53 46237137 IC50 > 12 ug.mL-1 T19244 CQX93F 46398805 IC50 > 10000 nM T19244 C9JA2C 46700789 IC50 = 2900 nM T19244 CJ2D3O 46701015 IC50 > 25000 nM T19244 CM04ZI 46701016 IC50 = 9830 nM T19244 C0JWP5 46701017 IC50 > 25000 nM T19244 C5H0MJ 46701086 IC50 > 25000 nM T19244 C9HWI7 46701087 IC50 > 25000 nM T19244 CVE5O1 46701088 IC50 > 25000 nM T19244 C1VPM0 46701089 IC50 > 25000 nM T19244 CQ8B6R 46701090 IC50 > 5000 nM T19244 C6C0FS 46701091 IC50 > 5000 nM T19244 C5TC2S 46830335 IC50 > 10000 nM T19244 C1K7FL 46830336 IC50 > 10000 nM T19244 C2M9XO 46835914 IC50 > 40000 nM T19244 C9CR0E 46835922 IC50 > 40000 nM T19244 C91HYQ 46840813 IC50 = 36 nM T19244 C1L0GS 46840949 IC50 = 83 nM T19244 C4C0ED 46840950 IC50 = 894 nM T19244 CI1YK3 46841216 IC50 = 2200 nM T19244 CD8M3F 46841499 IC50 = 264 nM T19244 CO76ID 46841501 IC50 = 184 nM T19244 CS5EJ1 46841648 IC50 = 17992 nM T19244 CRE97F 46841787 IC50 = 1101 nM T19244 COV0Q3 46841788 IC50 = 658 nM T19244 C2OWF8 46841789 IC50 = 552 nM T19244 C1N4KX 46842383 IC50 > 10000 nM T19244 CPE23Q 46850145 IC50 > 20000 nM T19244 C2UYK7 46850264 IC50 > 50000 nM T19244 CD04SA 46852212 IC50 > 3000 nM T19244 CT6MJ2 46852951 IC50 > 50000 nM T19244 CBZE98 46853681 IC50 > 30000 nM T19244 CO31WX 46861576 IC50 = 21900 nM T19244 C0EG8P 46865563 IC50 > 50000 nM T19244 C2P0SC 46865762 IC50 = 1440 nM T19244 C9T0ZE 46866390 IC50 < 300 nM T19244 CO3P0J 46866604 IC50 > 30000 nM T19244 C65BWF 46867649 IC50 > 10000 nM T19244 C8C3QD 46867792 IC50 > 10000 nM T19244 C1XGZ8 46867925 IC50 = 4110 nM T19244 CVH4G9 46867926 IC50 > 10000 nM T19244 CB6VI7 46867927 IC50 > 10000 nM T19244 C8OY4U 46869951 IC50 > 30000 nM T19244 C5I8ML 46871778 IC50 = 10200 nM T19244 C2LMI8 46871779 IC50 = 800 nM T19244 CLVI62 46879428 IC50 > 100000 nM T19244 CL2A4H 46879430 IC50 = 68000 nM T19244 C9VRO6 46879432 IC50 = 66000 nM T19244 CFH9W8 46879490 IC50 = 33000 nM T19244 CG68BI 46879549 IC50 = 3300 nM T19244 C9H1PK 46879550 IC50 = 6700 nM T19244 CB02YQ 46879551 IC50 = 1400 nM T19244 CCM7T2 46879552 IC50 = 61000 nM T19244 C7EHZ9 46879553 IC50 = 2300 nM T19244 CVI5O7 46879596 IC50 = 2700 nM T19244 CL05QN 46879597 IC50 = 700 nM T19244 CYK18D 46879598 IC50 = 11400 nM T19244 CG9N6P 46879643 IC50 = 500 nM T19244 CCK8A9 46880206 IC50 = 14000 nM T19244 C4BH9E 46882458 IC50 = 600 nM T19244 CERN34 46882461 IC50 = 2500 nM T19244 CRU1P2 46882874 IC50 < 10000 nM T19244 CYU8X6 46882875 IC50 > 10000 nM T19244 CX5CZ7 46882876 IC50 < 10000 nM T19244 C0FM2D 46882917 IC50 < 10000 nM T19244 CC1VO9 46882918 IC50 > 10000 nM T19244 C27RIV 46882919 IC50 > 10000 nM T19244 CE3O7D 46882949 IC50 < 10000 nM T19244 CHS1X0 46882950 IC50 < 10000 nM T19244 C3S9WE 46882951 IC50 > 10000 nM T19244 C3A1ZF 46882969 IC50 > 10000 nM T19244 CG3D0K 46882971 IC50 > 10000 nM T19244 CD7XA2 46882972 IC50 = 10000 nM T19244 CY5CW2 46882973 IC50 > 10000 nM T19244 C3ZPY7 46882986 IC50 > 10000 nM T19244 CKX8N2 46882987 IC50 > 10000 nM T19244 CG81CZ 46882988 IC50 > 10000 nM T19244 CP87CA 46883032 IC50 > 10000 nM T19244 CWU4T2 46883033 IC50 = 10000 nM T19244 C41RYD 46883034 IC50 > 10000 nM T19244 C3SQ2Z 46883035 IC50 > 10000 nM T19244 CS51UC 46883473 IC50 > 10000 nM T19244 CL0S4B 46883474 IC50 < 10000 nM T19244 C0K5ZJ 46883508 IC50 < 10000 nM T19244 CMNJ24 46883509 IC50 < 10000 nM T19244 CF4VC1 46883510 IC50 < 10000 nM T19244 CB8GE1 46884818 IC50 > 10000 nM T19244 C4MQ0A 46884856 IC50 > 10000 nM T19244 CCNT25 46884898 IC50 > 10000 nM T19244 C3MSG2 46885027 IC50 > 10000 nM T19244 CB7XI0 46885213 IC50 > 10000 nM T19244 CRE96X 46885625 IC50 < 100 nM T19244 CM76UZ 46888550 IC50 > 12 ug.mL-1 T19244 CX18GT 46889932 IC50 > 10000 nM T19244 C3C7OD 46890163 IC50 = 2500 nM T19244 CWSN39 46890164 IC50 = 15000 nM T19244 CVAU45 46890301 IC50 = 23000 nM T19244 C7QIT8 46891216 IC50 = 8100 nM T19244 CW7R5O 46891217 IC50 = 300 nM T19244 CSIX69 46891218 IC50 = 100 nM T19244 CZ90FC 46894119 IC50 = 1600 nM T19244 C90NYX 46896338 IC50 = 29000 nM T19244 CC9FZ0 46898063 IC50 > 20 nM T19244 C1JSH9 46899637 IC50 > 10000 nM T19244 CV3LP2 46899639 IC50 > 6000 nM T19244 CGHZ15 46899640 IC50 > 10000 nM T19244 CWR9M5 46900138 IC50 > 10000 nM T19244 CGN7Q8 46900139 IC50 > 10000 nM T19244 CN9FC3 46900150 IC50 = 4000 nM T19244 C40ZJO 46900451 IC50 < 4000 nM T19244 CNC02A 46900453 IC50 < 4000 nM T19244 CTCH14 46900455 IC50 < 4000 nM T19244 CP41AQ 46900457 IC50 < 2000 nM T19244 CR3L4I 46900459 IC50 > 10000 nM T19244 CK17PA 46900606 IC50 > 5000 nM T19244 C5ZT1B 46900610 IC50 = 4000 nM T19244 C1NAX4 46900612 IC50 > 5000 nM T19244 CT0SQ2 46900614 IC50 = 4000 nM T19244 CXD9S3 46900776 IC50 > 10000 nM T19244 C8I7SJ 46900778 IC50 = 2000 nM T19244 C7QDM9 46900782 IC50 > 8000 nM T19244 C15FMY 46900954 IC50 > 7000 nM T19244 C3JCB1 46911060 IC50 > 50000 nM T19244 C4WXU5 46911119 IC50 = 4300 nM T19244 C2YM9P 46911173 IC50 = 2400 nM T19244 CHUV97 46911229 IC50 > 5000 nM T19244 C1VA0B 46912953 IC50 > 5000 nM T19244 CLV1W2 46918487 IC50 > 10000 nM T19244 CJ3FM4 46925833 IC50 = 5030 nM T19244 CM8EH2 46926717 IC50 = 500 nM T19244 C65QAB 46927297 IC50 > 10000 nM T19244 C8GAI9 46927903 IC50 > 10000 nM T19244 CKO76R 46931815 IC50 > 5000 nM T19244 CV98OS 46933385 IC50 > 20000 nM T19244 C0J8WS 46933530 IC50 > 20000 nM T19244 CJK53D 46933697 IC50 = 9000 nM T19244 CU90MG 46938037 IC50 > 20000000 nM T19244 CX2U5I 46938097 IC50 > 20000000 nM T19244 C47QBL 46938101 IC50 > 20000000 nM T19244 C9DLV2 46945057 IC50 > 50000 nM T19244 CZ0G6A 46947062 IC50 = 43120 nM T19244 CX6NK2 47144386 IC50 = 24200 nM T19244 CBV0H3 49765039 IC50 = 3500 nM T19244 CWU2R3 49773361 IC50 > 40000 nM T19244 C9RI3L 49780809 IC50 > 4000 nM T19244 CYL65E 49781476 IC50 > 10000 nM T19244 CY1OJ5 49797177 IC50 > 30000 nM T19244 CZ2VI0 49797792 IC50 = 7943.28 nM T19244 CMY64F 49797816 IC50 = 10000 nM T19244 C8MH5L 49797817 IC50 = 19952.62 nM T19244 CF20IS 49797818 IC50 = 31622.78 nM T19244 C67IVU 49797819 IC50 = 39810.72 nM T19244 CUPE63 49797844 IC50 = 19952.62 nM T19244 CI2G9O 49797845 IC50 = 31622.78 nM T19244 CK5J8Z 49797846 IC50 = 10000 nM T19244 CW2VZ1 49797847 IC50 = 19952.62 nM T19244 CN6X3L 49797848 IC50 = 100 nM T19244 CH4KC8 49797849 IC50 = 15848.93 nM T19244 CWP4S9 49797850 IC50 = 79.43 nM T19244 CQVG17 49798349 IC50 = 4168.69 nM T19244 C62VRQ 49798437 IC50 = 5011.87 nM T19244 CY90CD 49798461 IC50 = 1348.96 nM T19244 CF8J6E 49798462 IC50 = 1071.52 nM T19244 C02EUQ 49800098 IC50 > 10000 nM T19244 CD8KX3 49804491 IC50 > 30000 nM T19244 CET89N 49822116 IC50 > 20000 nM T19244 CVS85M 49831162 IC50 = 5000 nM T19244 CA04IH 49836290 IC50 = 900 nM T19244 CDO7I4 49836293 IC50 = 4100 nM T19244 CT7CV0 49836295 IC50 > 10000 nM T19244 CYJW87 49836299 IC50 > 10000 nM T19244 C8E6WA 49836410 IC50 > 10000 nM T19244 CNM9X8 49836528 IC50 > 10000 nM T19244 COK75S 49836633 IC50 > 10000 nM T19244 CB81YG 49836637 IC50 > 10000 nM T19244 CD8GN9 49837170 EC50 = 22000 nM T19244 CB71TA 49837867 IC50 = 19000 nM T19244 CZQC64 49837869 IC50 = 14000 nM T19244 CVNA15 49837870 IC50 = 32000 nM T19244 C9L3XR 49838879 IC50 = 23000 nM T19244 C06MKW 49839561 IC50 > 10000 nM T19244 C3DN7U 49843520 IC50 = 280 nM T19244 CY46CB 49843532 IC50 > 50000 nM T19244 CU63QR 49847377 IC50 > 50000 nM T19244 CZT4I8 49847378 IC50 > 50000 nM T19244 CA72PE 49847379 IC50 > 50000 nM T19244 C8KQB9 49848139 IC50 > 10000 nM T19244 C4V7EW 49848258 IC50 > 10000 nM T19244 C4BXP1 49848557 IC50 > 50000 nM T19244 CHLR06 49848655 IC50 = 7943.28 nM T19244 CQ32CR 49848656 IC50 > 10000 nM T19244 C07NGT 49848778 IC50 = 5011.87 nM T19244 CP8TS6 49848895 IC50 > 50000 nM T19244 C9COF5 49848896 IC50 > 50000 nM T19244 CK0B1G 49848897 IC50 > 50000 nM T19244 C74KWB 49848898 IC50 = 3981.07 nM T19244 CP61VJ 49849002 IC50 > 50000 nM T19244 CBM62Z 49849007 IC50 > 50000 nM T19244 C05SEW 49849008 IC50 > 50000 nM T19244 CF64IJ 49849120 IC50 > 50000 nM T19244 CC9EB4 49849122 IC50 > 50000 nM T19244 C2ORV5 49849123 IC50 > 50000 nM T19244 CTR7Q0 49850345 IC50 > 50118.72 nM T19244 C8LBU5 49855513 IC50 > 30000 nM T19244 CQ0L4M 49856084 IC50 > 30000 nM T19244 C9TO2S 49856484 IC50 > 8900 nM T19244 CC8VZ4 49857811 IC50 > 30000 nM T19244 CZO5D6 49857998 IC50 > 30000 nM T19244 CXT41G 49862010 IC50 = 200 nM T19244 COS71Z 49862053 IC50 < 100 nM T19244 C4RNH2 49862091 IC50 = 200 nM T19244 CY9QB4 49862092 IC50 = 100 nM T19244 CC6NY3 49862093 IC50 = 1700 nM T19244 C6MP7Y 49862094 IC50 = 8900 nM T19244 CKO54S 49862127 IC50 = 700 nM T19244 C3O5IR 49862128 IC50 = 400 nM T19244 C9PCE3 49862155 IC50 >= 7000 nM T19244 CI41BU 49862643 IC50 = 100 nM T19244 C6O4ZK 49862647 IC50 > 5000 nM T19244 C10CAN 49862783 IC50 < 100 nM T19244 CGYM04 49864794 IC50 > 20000 nM T19244 CD29IW 49865043 IC50 > 20000 nM T19244 C0Y5ZU 49865137 IC50 > 20 nM T19244 CG98LM 49865191 IC50 = 2.6 nM T19244 C0S8XD 49865953 IC50 = 2600 nM T19244 CMV6Y2 49868651 IC50 > 40000 nM T19244 CCX18D 49871902 IC50 > 20000 nM T19244 CXI9D0 49871995 IC50 = 2000 nM T19244 C7GR0H 49872381 IC50 = 5660 nM T19244 CD1X3U 49872384 IC50 = 8510 nM T19244 C2ZG9D 49872391 IC50 = 640 nM T19244 C60RMP 49872483 IC50 = 12300 nM T19244 CS47WU 49872583 IC50 = 840 nM T19244 C83CTW 49872868 IC50 = 200 nM T19244 CY7QF8 49873368 IC50 = 340 nM T19244 CU7TK4 50899749 IC50 > 20000 nM T19244 CZ9UD6 50901657 IC50 > 50000 nM T19244 C1N4YP 50908737 IC50 > 10000 nM T19244 CENW12 50925404 IC50 = 20300 nM T19244 CMF7T6 50925457 IC50 > 5000 nM T19244 C2GTE4 50938548 IC50 > 50000 nM T19244 C4DH0A 50938549 IC50 = 9800 nM T19244 CJ43IF 50941460 IC50 > 25000 nM T19244 CLIK30 50941729 IC50 > 10000 nM T19244 CP7B9V 50942696 IC50 = 1800 nM T19244 CW6LP3 50992864 IC50 = 2000 nM T19244 C6UN8M 50992932 IC50 = 8000 nM T19244 C2SHO8 50993865 IC50 > 25000 nM T19244 CNBU93 50994740 IC50 < 3000 nM T19244 CH82SZ 51000500 IC50 = 24000 nM T19244 CX6PZ9 51003130 IC50 = 640 nM T19244 CAZQ43 51003133 IC50 = 6000 nM T19244 C8VNM2 51003549 IC50 > 50000 nM T19244 CP6NI2 51030711 IC50 > 30000 nM T19244 C70OGS 51030984 IC50 > 30000 nM T19244 CX28ZP 51030985 IC50 > 30000 nM T19244 CXB2Q6 51031001 IC50 > 30000 nM T19244 CUG03K 51033838 IC50 > 10000 nM T19244 C7OB2X 51035721 IC50 > 25000 nM T19244 CU1L3G 51038269 IC50 = 110 nM T19244 C96AQN 51346908 IC50 > 30000 nM T19244 CGW84J 51346919 IC50 > 50000 nM T19244 C3I7XR 51346964 IC50 > 10000 nM T19244 CD2YU8 51351496 IC50 = 3000 nM T19244 C2UG4W 51351504 IC50 = 4000 nM T19244 CAO41L 51351511 IC50 > 30000 nM T19244 CG3PR6 52912222 IC50 = 13000 nM T19244 CJ86KR 52917690 IC50 > 20000 nM T19244 CAXJ10 52918120 IC50 = 794.33 nM T19244 CRN19G 52918121 IC50 = 794.33 nM T19244 CTJ28K 52918135 IC50 = 29000 nM T19244 CJD25G 52920263 IC50 = 16000 nM T19244 CX9VO4 52932634 IC50 = 1300 nM T19244 C7VN1E 52934039 IC50 = 9800 nM T19244 CQ7EZ1 52934040 IC50 = 2300 nM T19244 CNOH36 52935183 IC50 = 1000 nM T19244 C10WZR 52940895 IC50 = 9400 nM T19244 C2RW5A 52940961 IC50 > 6000 nM T19244 CSXY62 52941059 IC50 > 30000 nM T19244 CQW15U 52941269 IC50 > 50000 nM T19244 C1YLX8 52941699 IC50 > 10000 nM T19244 C6NR7I 52942081 IC50 > 30000 nM T19244 C3BO1Z 52942119 IC50 = 8000 nM T19244 C34WMT 52942456 IC50 > 10000 nM T19244 CSHK08 52942937 IC50 = 3700 nM T19244 C3TK2O 52943442 IC50 > 30000 nM T19244 CTI28E 52944579 IC50 > 50000 nM T19244 CX0YD9 52944600 IC50 = 20000 nM T19244 CXTM57 52944645 IC50 = 11400 nM T19244 CHY9P7 52945359 IC50 = 2800 nM T19244 CO7ZR1 52947102 IC50 = 23100 nM T19244 C2YK4B 52947710 IC50 = 2400 nM T19244 CST08G 52947776 IC50 = 2100 nM T19244 CVF79G 52947777 IC50 = 3800 nM T19244 C56NDZ 52948169 IC50 = 2400 nM T19244 C48JMX 52948255 IC50 > 50000 nM T19244 C7SAC6 52948857 IC50 > 10000000 nM T19244 C43KTX 52948925 IC50 = 4100 nM T19244 C0HA6F 52949188 IC50 = 3700 nM T19244 C3DTV5 53233133 IC50 > 10000 nM T19244 C2RCZ0 53235503 IC50 > 20000 nM T19244 C9RIJ7 53237893 IC50 = 34000 nM T19244 C5ZT7N 53237897 IC50 = 40000 nM T19244 C4KRV8 53237899 IC50 = 40000 nM T19244 C0H6TR 53237903 IC50 = 34000 nM T19244 CIP64Q 53238125 IC50 = 40000 nM T19244 C2AUL9 53248760 IC50 > 50000 nM T19244 CP3J9M 53248845 IC50 > 50000 nM T19244 CQIY23 53248846 IC50 > 50000 nM T19244 C9MHR0 53248847 IC50 = 28000 nM T19244 CT9V3I 53251325 IC50 = 81600 nM T19244 CY28CB 53257408 EC50 = 3981.07 nM T19244 CL62UR 53257683 IC50 > 3000 nM T19244 CFJT89 53260268 EC50 = 15848.93 nM T19244 CX69QK 53260269 EC50 = 25118.86 nM T19244 CD35QU 53308640 IC50 > 10000 nM T19244 CRI92N 53311230 IC50 > 10000 nM T19244 CQ9HO5 53311701 IC50 = 1300 nM T19244 CL78NK 53316823 IC50 > 25000 nM T19244 C1-MAY-02 53317017 IC50 > 50000 nM T19244 CK27PC 53317643 IC50 = 40000 nM T19244 CXV3W2 53317718 IC50 = 21000 nM T19244 CP14EK 53317957 IC50 = 13600 nM T19244 CL45CT 53318503 IC50 > 5000 nM T19244 C5F1IR 53318745 IC50 = 25000 nM T19244 CZ0M8J 53319021 IC50 > 10000 nM T19244 COJ82D 53319320 IC50 = 6400 nM T19244 CK2G3D 53319480 IC50 > 25000 nM T19244 C90TZS 53319482 IC50 > 10000 nM T19244 CTA23R 53319654 IC50 = 18000 nM T19244 CXY8A4 53319905 IC50 > 38000 nM T19244 CXF1S4 53320328 IC50 > 25000 nM T19244 CB84NG 53320778 IC50 > 25000 nM T19244 C5HL4R 53321372 IC50 > 25000 nM T19244 C4X3IS 53321979 IC50 > 25000 nM T19244 CLD82J 53322084 IC50 > 25000 nM T19244 CY09UA 53322086 IC50 = 7600 nM T19244 CBUT35 53322087 IC50 > 10000 nM T19244 CMH54U 53322279 IC50 > 50000 nM T19244 CR57HN 53323639 IC50 = 6700 nM T19244 CX54CT 53323813 IC50 > 25000 nM T19244 CC08MY 53324265 IC50 = 28000 nM T19244 CC1ER2 53324598 IC50 = 18000 nM T19244 C3QNR2 53325463 IC50 > 25000 nM T19244 CZN8B4 53325581 IC50 > 25000 nM T19244 CZ1SE0 53325908 IC50 = 4200 nM T19244 C1N7XO 53325966 IC50 = 250 nM T19244 C28HNA 53326213 IC50 = 7100 nM T19244 C18TPG 53326909 IC50 > 25000 nM T19244 C7J8ZY 53327611 IC50 = 1900 nM T19244 C8PJ6E 53354789 IC50 = 3000 nM T19244 CYMP74 53354793 IC50 = 23000 nM T19244 C8ZRE3 53356518 IC50 = 400 nM T19244 CL89US 53359023 IC50 > 50000 nM T19244 CRZL59 53361076 IC50 > 40000 nM T19244 C9H5YE 53361128 IC50 = 4900 nM T19244 CC7DZ4 53362086 IC50 > 50000 nM T19244 CX83CK 53362097 IC50 > 8900 nM T19244 C1F8IK 53363810 IC50 > 30000 nM T19244 C9GYZ3 53372790 IC50 = 8700 nM T19244 CT6K2O 53373472 IC50 = 27000 nM T19244 CL37YO 53380288 IC50 > 10000 nM T19244 C1Q0OJ 53382545 IC50 > 30000 nM T19244 C19HFO 53386426 IC50 = 7900 nM T19244 CZWO31 53387025 IC50 > 100000 nM T19244 C7KM5B 53388319 IC50 = 1 nM T19244 CIGM78 53389570 IC50 > 30000 nM T19244 C64TJO 53391717 IC50 > 25000 nM T19244 C3Q6IL 53391718 IC50 = 14400 nM T19244 C6AYE3 53392451 IC50 > 100000 nM T19244 C47VGW 53393916 IC50 > 30000 nM T19244 C24FQU 53465297 IC50 > 12000 nM T19244 C0T5VA 53467975 IC50 > 11000 nM T19244 C2XHO3 53468206 IC50 > 11000 nM T19244 CX0R1K 53469059 IC50 = 24700 nM T19244 CV7C0D 53469060 IC50 = 19200 nM T19244 CCKD45 53469061 IC50 > 25000 nM T19244 C3SRN7 53469411 IC50 = 1330 nM T19244 CK1C9O 53472113 IC50 = 3000 nM T19244 CITN21 53475321 IC50 > 20000 nM T19244 C9EF7S 53482945 IC50 = 66000 nM T19244 CFU8T7 53483937 IC50 > 30000 nM T19244 CG3FA9 53492750 IC50 = 4300 nM T19244 C4U5IX 53493001 IC50 > 35000 nM T19244 CE9K7U 53494972 IC50 > 10000 nM T19244 C7TR2W 53497131 IC50 = 21000 nM T19244 CGSN74 53497490 IC50 = 11500 nM T19244 CVA4I0 54576291 IC50 > 10000 nM T19244 CSAV94 54576503 IC50 > 10000 nM T19244 COF6B0 54577892 IC50 > 30000 nM T19244 C2ECL9 54577896 IC50 > 30000 nM T19244 CP24ZC 54579002 IC50 = 4400 nM T19244 C7FXV6 54580144 IC50 = 26000 nM T19244 CRB0W3 54580721 IC50 > 50000 nM T19244 C2XV8F 54581365 IC50 = 1500 nM T19244 C2RJM1 54583706 IC50 > 50000 nM T19244 CHP62C 54584119 IC50 = 13000 nM T19244 C37TZQ 54584868 IC50 > 30000 nM T19244 CQ0G6R 54586630 IC50 = 2400 nM T19244 CQWI92 54586805 IC50 > 30000 nM T19244 CXU62W 54677935 IC50 > 40000 nM T19244 CXH5O8 54681545 Ki = 500 nM T19244 C0ZG2V 54709839 IC50 > 100000 nM T19244 C47XPL 54710283 Ki = 3000 nM T19244 CWQ1J8 54710483 Ki = 1100 nM T19244 CO75TL 54712015 IC50 > 50000 nM T19244 CLT3Q8 54716246 IC50 = 75000 nM T19244 CVHT05 54723704 Ki = 100 nM T19244 C1Z3SX 54723890 Ki = 3000 nM T19244 C98BDH 54724723 Ki = 1500 nM T19244 C91XGI 54736486 Ki = 400 nM T19244 CMN1C6 54752118 IC50 > 10000 nM T19244 CZY7F9 54752621 IC50 > 7000 nM T19244 C69EQM 54752774 IC50 > 10000 nM T19244 CD8YN4 54753626 IC50 > 30000 nM T19244 CL32AY 54753627 IC50 > 30000 nM T19244 CBO2L1 54761157 IC50 > 40000 nM T19244 C0Y9ZG 54761473 IC50 > 10000 nM T19244 CS23GM 54762055 IC50 > 40000 nM T19244 CPS5V6 54764158 IC50 > 30000 nM T19244 C0T3KY 54765285 IC50 > 11000 nM T19244 CJ9B4P 54768039 IC50 > 10000 nM T19244 C79DVG 56589615 IC50 > 30000 nM T19244 C23NQS 56593147 IC50 > 20000 nM T19244 CXSQ19 56593712 IC50 = 72700 nM T19244 CHD79F 56594864 IC50 = 1700 nM T19244 CMQ2J3 56594865 IC50 > 10000 nM T19244 C6FE3Z 56594866 IC50 > 10000 nM T19244 CS3E5I 56594867 IC50 > 10000 nM T19244 C91PGO 56603115 IC50 > 50000 nM T19244 C5ES6P 56603116 IC50 = 10800 nM T19244 CVI51O 56603118 IC50 > 50000 nM T19244 C2IM6T 56603174 IC50 > 50000 nM T19244 CH05TN 56603175 IC50 > 50000 nM T19244 CDL94H 56603301 IC50 = 20400 nM T19244 C9D1MV 56603353 IC50 = 39500 nM T19244 CJVR02 56603413 IC50 = 3400 nM T19244 C9ZF6B 56643412 IC50 > 25000 nM T19244 CQ18BI 56643478 IC50 = 10000 nM T19244 CBJ4V8 56649677 IC50 = 9900 nM T19244 CPJ7D3 56658546 IC50 > 30000 nM T19244 C7AG6I 56658547 IC50 > 30000 nM T19244 C6W5UT 56658548 IC50 > 30000 nM T19244 C9TFO2 56658589 IC50 = 1000 nM T19244 CFT9V8 56659147 IC50 > 25000 nM T19244 CGID30 56659201 IC50 > 10000 nM T19244 C2QTH5 56662000 IC50 > 30000 nM T19244 CC1GK4 56665357 IC50 > 30000 nM T19244 C25HCW 56668953 IC50 = 1000 nM T19244 CC9XR7 56669562 IC50 > 10000 nM T19244 CXE9A8 56669563 IC50 > 8000 nM T19244 C9MW0X 56670034 IC50 < 10000 nM T19244 CK9L4C 56672570 IC50 > 30000 nM T19244 CKVS08 56676902 IC50 = 350 nM T19244 CZP86D 56677285 IC50 > 30000 nM T19244 C7QW5F 56678507 IC50 > 10000 nM T19244 CW7QF9 56679101 IC50 > 30000 nM T19244 CUIB93 56679632 IC50 = 141000 nM T19244 CK73UC 56683046 IC50 > 6000 nM T19244 CJC19B 56683709 IC50 > 30000 nM T19244 CY3G8F 56834936 IC50 = 700 nM T19244 CR7LS4 56835090 IC50 > 30000 nM T19244 C70GHX 56835991 IC50 > 50000 nM T19244 CH2AY6 56838673 IC50 = 4000 nM T19244 C3OE8N 56838888 IC50 > 30000 nM T19244 CY6UB2 56839590 IC50 = 1700 nM T19244 CVYF04 56840671 IC50 > 10000 nM T19244 CR8KU2 56840672 IC50 > 10000 nM T19244 C7CWA4 56842683 Ki = 3000 nM T19244 CKY51C 56847605 IC50 = 54000 nM T19244 CUY28J 56850524 IC50 = 12 nM T19244 CK0I6Q 56850525 IC50 = 1.5 nM T19244 C1U7XJ 56924869 IC50 > 30000 nM T19244 CZRQ14 56929159 IC50 = 54000 nM T19244 C9IVD0 56929216 IC50 > 10000 nM T19244 C90URY 56929249 IC50 = 54000 nM T19244 CPAU51 56943206 IC50 = 54 nM T19244 CI04WC 56948248 IC50 = 15500 nM T19244 CL16UQ 56949326 IC50 = 3500 nM T19244 C71JRF 56949451 IC50 = 300 nM T19244 C89PEN 56949822 IC50 > 10000 nM T19244 C1K8TD 56949966 IC50 > 10000 nM T19244 CWB5H7 56953768 IC50 = 9180 nM T19244 CS0HF1 56953769 IC50 = 2920 nM T19244 CPJ7X3 56953770 IC50 = 4570 nM T19244 CK7M6W 56953771 IC50 = 21200 nM T19244 CO96BR 56953896 IC50 = 22100 nM T19244 CJ0WM6 56953897 IC50 = 4410 nM T19244 C4UV1D 56953898 IC50 = 3420 nM T19244 CPKI96 56954010 IC50 = 5150 nM T19244 C6Q8BZ 56954011 IC50 = 820 nM T19244 C5G4UX 56954012 IC50 = 6180 nM T19244 C8UQ2S 56954013 IC50 = 960 nM T19244 CHQA53 56954137 IC50 = 880 nM T19244 CZGE53 56954138 IC50 = 22300 nM T19244 CGRC25 56954242 IC50 < 205 nM T19244 CRT0Y2 56954243 IC50 = 213 nM T19244 CAK91L 56955954 IC50 = 591 nM T19244 CD3SZ1 56959836 IC50 = 2400 nM T19244 CN2GI7 56959991 IC50 = 560 nM T19244 CKN0Z8 56964577 IC50 > 25000 nM T19244 CS7U9L 56965952 IC50 = 1000 nM T19244 CT67IO 57325589 IC50 > 25000 nM T19244 CV5CP4 57326678 IC50 = 4300 nM T19244 CLB5K0 57331386 IC50 > 10000 nM T19244 CGUA26 57331668 IC50 > 50000 nM T19244 CFW0D1 57339435 IC50 = 10000 nM T19244 C4G7QD 57343225 IC50 = 9000 nM T19244 CT8VZ6 57345658 IC50 > 30000 nM T19244 C7O0AI 57345659 IC50 > 30000 nM T19244 C3L9ZA 57345660 IC50 > 30000 nM T19244 CZK3M1 57345661 IC50 > 30000 nM T19244 C34DJP 57384236 IC50 > 50000 nM T19244 CEOC15 57384237 IC50 > 50000 nM T19244 CY50WC 57384238 IC50 = 25000 nM T19244 C7S0ZR 57384239 IC50 = 30000 nM T19244 C2XN1G 57384481 IC50 = 10000 nM T19244 CR73IZ 57384482 IC50 > 50000 nM T19244 CR2M5H 57384483 IC50 = 44000 nM T19244 CQ72HI 57384749 IC50 > 50000 nM T19244 C68KGE 57384750 IC50 > 50000 nM T19244 CCT5D4 57386783 IC50 > 50000 nM T19244 CC30XZ 57386784 IC50 > 50000 nM T19244 C79BXP 57386785 IC50 > 50000 nM T19244 CM6DV7 57387028 IC50 > 50000 nM T19244 C0GS4F 57387282 IC50 > 50000 nM T19244 C0TL9C 57387283 IC50 > 50000 nM T19244 CAU3G9 57387540 IC50 > 50000 nM T19244 CL2AO8 57387541 IC50 > 50000 nM T19244 C0XWL8 57387542 IC50 > 50000 nM T19244 CC4DK0 57387775 IC50 > 50000 nM T19244 C56ORS 57388650 IC50 > 10000 nM T19244 C5OJP0 57391102 IC50 > 25000 nM T19244 CR8MW2 57391205 IC50 > 10000 nM T19244 CNQ9B2 57392969 IC50 > 10000 nM T19244 C04IST 57394707 IC50 > 10000 nM T19244 CNOH63 57394711 IC50 > 10000 nM T19244 C6HBG0 57396813 IC50 > 30000 nM T19244 CU4FW8 57397383 IC50 > 25000 nM T19244 CQS0M5 57397654 IC50 > 30000 nM T19244 C4RHF3 57404027 IC50 > 30000 nM T19244 C6XA7G 57405264 IC50 > 30000 nM T19244 CUOV05 57411066 IC50 > 30000 nM T19244 CM3T2V 57431767 IC50 = 2400 nM T19244 C8LVD4 57431775 IC50 = 2400 nM T19244 CI4V2N 57431852 IC50 = 7000 nM T19244 C0MBP3 57431914 IC50 = 16000 nM T19244 C9ZMQ1 57480972 IC50 = 7000 nM T19244 COUZ63 57494822 IC50 = 372 nM T19244 C37SMZ 57505249 IC50 = 55000 nM T19244 C23FTC 57510027 IC50 > 20000 nM T19244 C7I4QD 57519510 IC50 > 50000 nM T19244 C3N4MF 57520842 IC50 > 50000 nM T19244 CEL56T 57520942 IC50 > 50000 nM T19244 C1HRZ7 57544434 IC50 = 900 nM T19244 C7D1JL 57606048 IC50 = 7000 nM T19244 CSD0M2 57658880 IC50 = 11000 nM T19244 CIFW58 57658935 IC50 = 14000 nM T19244 CV2J9A 57663655 IC50 = 51000 nM T19244 CTM6K5 57690900 IC50 = 17000 nM T19244 C35GXV 57720515 EC50 > 40000 nM T19244 C58TKU 57773771 IC50 > 25000 nM T19244 CY4O6Z 57965013 IC50 > 6000 nM T19244 CP28UL 57965039 IC50 > 25000 nM T19244 CANZ90 57994936 IC50 > 20000 nM T19244 CGBY54 58063225 IC50 > 10000 nM T19244 C0P8VW 58063334 IC50 > 5000 nM T19244 CZO2J1 58063487 IC50 > 10000 nM T19244 CSC1K6 58109236 IC50 = 33000 nM T19244 CS05MK 58109240 IC50 > 50000 nM T19244 CDC28F 58109250 IC50 > 50000 nM T19244 C4E2RC 58109371 IC50 = 22200 nM T19244 C4SC0Z 58109674 IC50 > 50000 nM T19244 C1EF0B 58109729 IC50 = 21400 nM T19244 CBZX94 58199027 IC50 > 30000 nM T19244 CB72QI 58204997 IC50 > 10000 nM T19244 C93STQ 58239274 IC50 > 20000 nM T19244 C2SE1Z 58239287 IC50 > 20000 nM T19244 CI45ZP 58269513 IC50 = 7000 nM T19244 CK10DA 58269516 IC50 = 8000 nM T19244 CV9FC4 58269518 IC50 = 29000 nM T19244 CM1GN4 58269523 IC50 = 16000 nM T19244 CAY0H7 58269562 IC50 > 30000 nM T19244 CN13SI 58269563 IC50 > 30000 nM T19244 CPQ0Z4 58269588 IC50 = 25000 nM T19244 C8A3JQ 58269598 IC50 = 7000 nM T19244 CD18IU 58269609 IC50 = 19000 nM T19244 CQV75S 58269620 IC50 = 4000 nM T19244 C26OPT 58269625 IC50 = 13000 nM T19244 C8ILS3 58269629 IC50 = 17000 nM T19244 C5VFQ7 58269655 IC50 = 13000 nM T19244 CQ63WZ 58269663 IC50 = 25000 nM T19244 C2PYB1 58269668 IC50 = 18000 nM T19244 CI3P0D 58269670 IC50 = 3000 nM T19244 C5RF8T 58269685 IC50 = 4000 nM T19244 C4OS3J 58269689 IC50 = 400 nM T19244 C3CFB8 58269691 IC50 = 21000 nM T19244 CZA32V 58344912 IC50 > 10000 nM T19244 CPVF85 58344916 IC50 > 10000 nM T19244 CY62SG 58345029 IC50 > 10000 nM T19244 CMXC37 58365250 IC50 = 18000 nM T19244 C4EPA5 58365345 IC50 = 8000 nM T19244 CO53TZ 58365501 IC50 > 20000 nM T19244 CXY58G 58365527 IC50 > 20000 nM T19244 CON6K1 58365686 IC50 = 18000 nM T19244 CVP17Q 58365704 IC50 > 20000 nM T19244 CZ6X0Y 58365744 IC50 = 18000 nM T19244 CX8Y6Z 58365813 IC50 = 5000 nM T19244 C3WB9I 58365828 IC50 = 8000 nM T19244 C5CRB1 58365867 IC50 = 8000 nM T19244 CF6A8Y 58365941 IC50 = 17000 nM T19244 C35RYZ 58365945 IC50 = 13000 nM T19244 CJI25C 58365995 IC50 = 9000 nM T19244 C3QI6Y 58366053 IC50 = 15000 nM T19244 C6AC9L 58366064 IC50 = 4000 nM T19244 CC67BX 58366073 IC50 > 20000 nM T19244 C0F3BO 58394783 IC50 > 10000 nM T19244 C0X7IK 58394837 IC50 > 10000 nM T19244 CASI81 58395078 IC50 > 10000 nM T19244 CWBM72 58395283 IC50 > 10000 nM T19244 C6BZ0G 58439416 IC50 = 11000 nM T19244 CAW51G 58486138 IC50 = 1700 nM T19244 CRB42N 58486297 IC50 = 3800 nM T19244 C35FWX 58486367 IC50 > 10000 nM T19244 C6JKM0 58834906 IC50 > 100000 nM T19244 CF9Z0L 58834953 IC50 > 26000 nM T19244 C4PWA9 58835024 IC50 > 40000 nM T19244 CCR4T7 58835217 IC50 > 73000 nM T19244 C9ZE7J 58874273 IC50 > 50000 nM T19244 C7CE6L 58950132 IC50 = 2500 nM T19244 C6ZQ3C 58973420 IC50 = 660 nM T19244 CCQM76 59153288 IC50 > 50000 nM T19244 C3L4JY 59176329 IC50 > 10000 nM T19244 C0U1HA 59179260 IC50 = 5620 nM T19244 CK7T6D 59179887 IC50 = 7860 nM T19244 C6DG2S 59190464 IC50 > 1000 nM T19244 CL9R5M 59190503 IC50 > 1000 nM T19244 CQHS47 59190547 IC50 > 1000 nM T19244 C79GHB 59190548 IC50 > 1000 nM T19244 CJ6R8Q 59251679 IC50 > 25000 nM T19244 C2PJ4N 59271992 IC50 > 20000 nM T19244 CUE79I 59272004 IC50 > 10000 nM T19244 C19YVT 59377518 IC50 > 32000 nM T19244 C1JK7V 59377559 IC50 > 50000 nM T19244 CFDG19 59401765 IC50 > 30000 nM T19244 CC5QW1 59401793 IC50 > 30000 nM T19244 CNOI48 59401886 IC50 > 30000 nM T19244 CJ2Y3A 59414201 IC50 = 8000 nM T19244 CN1US8 59447733 IC50 = 25000 nM T19244 C9S4DU 59447737 IC50 = 9600 nM T19244 CVZ09Q 59454159 IC50 = 4000 nM T19244 CK6LX0 59454220 IC50 = 13000 nM T19244 C2SDN1 59454252 IC50 = 23000 nM T19244 CK6W7I 59536635 IC50 > 10000 nM T19244 CA9NE4 59548712 IC50 > 30000 nM T19244 CM1G2P 59568656 IC50 > 50000 nM T19244 CS80HW 59648012 IC50 > 30000 nM T19244 C3RB0E 59648133 IC50 > 50000 nM T19244 CYKF93 59651916 IC50 > 30000 nM T19244 C5PDB3 59651957 IC50 > 30000 nM T19244 C4W8RH 59651989 IC50 > 30000 nM T19244 CBEG02 59721267 IC50 = 13400 nM T19244 CV6L5Y 59721273 IC50 > 25000 nM T19244 CS5U7D 59721308 IC50 > 25000 nM T19244 CK2UR9 59721409 IC50 = 4700 nM T19244 C4I3JA 59721419 IC50 = 4700 nM T19244 C7ECU2 59794447 IC50 > 40000 nM T19244 C5QS4J 60148513 IC50 = 4200 nM T19244 CK5N4E 60148693 IC50 = 400 nM T19244 C6L4RH 60148695 IC50 = 23000 nM T19244 CUYB59 60148924 IC50 = 1980 nM T19244 C4MV2N 60149678 IC50 > 30000 nM T19244 CTL97W 60151476 IC50 > 45000 nM T19244 C62SQG 60155628 IC50 = 100 nM T19244 COS39T 60155629 IC50 < 1000 nM T19244 CE5A7B 60162406 IC50 > 100000 nM T19244 C2D3HQ 60168069 IC50 = 12100 nM T19244 CIJ16Y 60196616 IC50 = 21500 nM T19244 C3S1RP 60197614 IC50 = 4100 nM T19244 CS4F2O 60197712 IC50 > 30000 nM T19244 C87HTO 60197713 IC50 = 1800 nM T19244 C5ES4W 60197714 IC50 = 11000 nM T19244 CF19XN 60197716 IC50 > 30000 nM T19244 COI61M 60197822 IC50 = 1300 nM T19244 CP1CK0 60197823 IC50 = 5700 nM T19244 C0JL3I 60197824 IC50 > 30000 nM T19244 CVOF90 60197825 IC50 = 1800 nM T19244 CBN3G4 60197937 IC50 = 1800 nM T19244 CT26JV 60202329 IC50 > 50000 nM T19244 CWA0B6 60204017 IC50 > 30000 nM T19244 CW3H0V 60634975 IC50 > 25000 nM T19244 C4BZ2N 60637368 IC50 > 25000 nM T19244 CV13OQ 62705051 IC50 > 40000 nM T19244 C9F4JW 62705832 IC50 < 2500 nM T19244 CJ5HI6 66547425 IC50 < 1000 nM T19244 CH76RD 66550504 IC50 > 25000 nM T19244 C2LBW7 66551925 IC50 > 50000 nM T19244 CLHX28 66553128 IC50 > 20000 nM T19244 CNDH38 66557868 IC50 > 10000 nM T19244 CUC7B3 66557964 IC50 > 30000 nM T19244 C23NWU 66562843 IC50 > 20000 nM T19244 CE2S6P 66562938 IC50 > 20000 nM T19244 CK9FO4 66562947 IC50 > 20000 nM T19244 C1WXS5 66563037 IC50 > 20000 nM T19244 CG34JD 66563137 IC50 > 20000 nM T19244 C6LVU1 66563478 IC50 > 20000 nM T19244 C7FX5M 66563570 IC50 > 20000 nM T19244 C24BOR 66563571 IC50 > 20000 nM T19244 CQY3J2 66563572 IC50 > 20000 nM T19244 CC6RH8 66574514 IC50 = 25700 nM T19244 CY81CB 66575661 IC50 = 9500 nM T19244 CMXA10 66575743 IC50 > 50000 nM T19244 CZF76R 66608383 IC50 > 30000 nM T19244 CJQ1K5 66610067 IC50 = 68 nM T19244 CRG3E9 66610246 IC50 = 200 nM T19244 C1W6FK 66610365 IC50 = 750 nM T19244 CS72TK 66610926 IC50 > 10000 nM T19244 CA2H3P 66611008 IC50 = 1050 nM T19244 CVB4T1 66611375 IC50 = 420 nM T19244 CUP41L 66613450 IC50 = 14800 nM T19244 CFI5T8 66613669 IC50 = 70 nM T19244 CY9TD4 66730677 IC50 > 10000 nM T19244 CJFS84 66731186 IC50 > 10000 nM T19244 CG1O8H 66734740 IC50 > 10000 nM T19244 C8CLK2 66735127 IC50 > 10000 nM T19244 CL5GH9 66735487 IC50 > 10000 nM T19244 CKN2U0 66764813 IC50 > 30000 nM T19244 C51XCV 66781377 IC50 > 10000 nM T19244 CU6E0A 66818541 IC50 > 30000 nM T19244 CKD8I1 66818569 IC50 > 30000 nM T19244 C5LU1Z 66818766 IC50 > 30000 nM T19244 C5J4MR 66850717 IC50 > 10000 nM T19244 CN7E8B 66853985 IC50 = 7400 nM T19244 C7A2EI 66854102 IC50 = 290 nM T19244 C32ADF 66895517 IC50 = 5700 nM T19244 C40FKD 66898172 IC50 > 50000 nM T19244 C7TJ9X 66898814 IC50 > 50000 nM T19244 CX1P8I 67042254 IC50 > 25000 nM T19244 CFM6H7 67049587 IC50 > 100000 nM T19244 C4NX6W 67070065 IC50 > 50000 nM T19244 CN8AS7 67072266 IC50 < 200000 nM T19244 CVT35R 67097557 IC50 = 2400 nM T19244 CJV8O4 67098558 IC50 = 3500 nM T19244 CE49GC 67098566 IC50 = 4900 nM T19244 COD28B 67098794 IC50 = 1400 nM T19244 C52XBW 67098971 IC50 < 200 nM T19244 CX6SF2 67250226 IC50 = 8500 nM T19244 CY76UR 67305743 IC50 = 7900 nM T19244 C3UKG8 67312397 IC50 = 1000 nM T19244 CM6TZ3 67312506 IC50 = 10000 nM T19244 CKMV48 67345882 IC50 > 10000 nM T19244 C50IMJ 67387021 IC50 > 20000 nM T19244 C4R8OG 67401728 IC50 > 30000 nM T19244 CX8JP5 67402849 IC50 > 40000 nM T19244 CPV39L 67406727 IC50 > 30000 nM T19244 C4S3FE 67450880 IC50 = 19000 nM T19244 C8L5HO 67453320 IC50 > 100000 nM T19244 CNB15W 67607112 IC50 = 8430 nM T19244 CE94JQ 67953283 IC50 = 46000 nM T19244 CT43SM 67953330 IC50 = 17000 nM T19244 CPTA39 67953837 IC50 > 50000 nM T19244 CAF36T 67972044 IC50 = 1800 nM T19244 C5K7QG 67974411 IC50 >= 30000 nM T19244 CO75NL 68011817 IC50 > 10000 nM T19244 CBOF40 68046989 IC50 = 35100 nM T19244 C02LWX 68074963 IC50 = 7000 nM T19244 CGW5L9 68075088 IC50 = 6000 nM T19244 CN3KZ8 68161075 IC50 = 14000 nM T19244 C3K4RT 68204896 IC50 < 10000 nM T19244 C32TVX 68230798 IC50 = 1700 nM T19244 C5YCB6 68234668 IC50 = 170 nM T19244 CR17ZU 68234693 IC50 = 190 nM T19244 CZCP37 68234870 IC50 = 140 nM T19244 C9J8GY 68234878 IC50 = 260 nM T19244 CN6KL0 68235029 IC50 = 570 nM T19244 C1KAG4 68235232 IC50 > 40000 nM T19244 C7TR4I 68276577 IC50 = 70 nM T19244 CD68FL 68277248 IC50 = 60 nM T19244 CK5V3O 68277611 IC50 = 200 nM T19244 CBV34D 68277935 IC50 = 50 nM T19244 C17JAZ 68284084 IC50 = 3400 nM T19244 CW70TJ 68284602 IC50 = 2500 nM T19244 CYCN51 68284666 IC50 > 10000 nM T19244 CW21KG 68284716 IC50 > 10000 nM T19244 CCT07V 68290289 IC50 > 20000 nM T19244 C4LKB3 68291752 IC50 > 20000 nM T19244 CPA95O 68380152 IC50 > 30000 nM T19244 C95VPL 68380260 IC50 = 15400 nM T19244 CVM9Q1 68503758 IC50 = 16000 nM T19244 CLS10P 68513301 IC50 = 7700 nM T19244 C5JYB8 68515257 IC50 = 18100 nM T19244 C69OHY 68560854 IC50 = 2000 nM T19244 CCD89X 68563058 IC50 = 30000 nM T19244 C48EIQ 68568011 IC50 = 600 nM T19244 CH3Z7F 68658979 IC50 > 50000 nM T19244 C89CQS 68779277 IC50 = 8600 nM T19244 CJI32G 69081964 IC50 > 30000 nM T19244 C02UFD 69224054 IC50 > 18000 nM T19244 C7SQT4 69224555 IC50 = 20000 nM T19244 C7Z9LF 69224988 IC50 = 15000 nM T19244 COJ4Q1 69315206 IC50 = 24000 nM T19244 CJ5Z7T 69316129 IC50 = 6000 nM T19244 C5VJG4 69643233 IC50 > 30000 nM T19244 CHD80I 69937162 IC50 > 50000 nM T19244 CAR2N8 69937236 IC50 > 50000 nM T19244 CN7X0U 69937257 IC50 > 50000 nM T19244 CC8QU9 70227534 IC50 = 4640 nM T19244 C06WFN 70276830 IC50 > 31622.78 nM T19244 CDQ85E 70276990 IC50 = 7943.28 nM T19244 CK5H1Y 70497007 IC50 > 10000 nM T19244 C6NSG3 70497750 IC50 > 10000 nM T19244 CWP52K 70497865 IC50 > 10000 nM T19244 C7VJ6A 70647728 IC50 > 8000 nM T19244 CFH68K 70664065 IC50 = 2400 nM T19244 CAR46Z 70675172 IC50 > 25000 nM T19244 CN09DI 70675846 IC50 = 4000 nM T19244 C97WSO 70678458 IC50 > 30000 nM T19244 CC6T5K 70679283 IC50 > 30000 nM T19244 C0I7PG 70681152 IC50 > 33000 nM T19244 C7GJW9 70681170 IC50 = 600 nM T19244 CAO1N7 70681171 IC50 = 1200 nM T19244 CC20VE 70681172 IC50 = 2200 nM T19244 C8H4JX 70681173 IC50 = 2800 nM T19244 C6NYK2 70681174 IC50 = 900 nM T19244 C7W3JA 70681326 IC50 > 5000 nM T19244 C8XC1S 70682487 IC50 > 20000 nM T19244 CPF92N 70682528 IC50 = 9500 nM T19244 C37CFL 70682529 IC50 = 9800 nM T19244 C8KBJ0 70683271 IC50 = 4300 nM T19244 CZHB48 70684601 IC50 = 2400 nM T19244 C5P0CI 70684602 IC50 = 14000 nM T19244 C86ETQ 70684603 IC50 = 10000 nM T19244 CCM9Z5 70684604 IC50 > 20000 nM T19244 C4FH7S 70684606 IC50 > 20000 nM T19244 CHFM92 70685176 IC50 > 50000 nM T19244 CG6BY1 70685177 IC50 > 30000 nM T19244 CWIC42 70685308 IC50 > 10000 nM T19244 CU50BK 70685377 IC50 = 5100 nM T19244 C3MB6V 70685378 IC50 = 8500 nM T19244 C60SBP 70685515 IC50 > 9000 nM T19244 CYO5N3 70686766 IC50 >= 5000 nM T19244 C4VU7J 70688210 IC50 > 50000 nM T19244 CQ0ZN8 70688528 IC50 = 3981.07 nM T19244 CZC4Y2 70688845 IC50 = 5600 nM T19244 CE1GI4 70688847 IC50 = 8300 nM T19244 C18OFS 70688848 IC50 > 20000 nM T19244 CIF26X 70689554 IC50 = 2100 nM T19244 C4GXP2 70690453 IC50 > 30000 nM T19244 C10XER 70691455 Ki = 140000 nM T19244 CH34MZ 70691697 IC50 = 700 nM T19244 CXD3F9 70691699 IC50 = 1200 nM T19244 C0XRC9 70691981 IC50 > 8600 nM T19244 C7UNV3 70692732 IC50 = 1584.89 nM T19244 CJ0P9G 70693067 IC50 = 7400 nM T19244 C8IOC9 70693068 IC50 = 7100 nM T19244 CF5YQ9 70693069 IC50 = 6800 nM T19244 CI4KP9 70693070 IC50 > 20000 nM T19244 CG4S9N 70693071 IC50 = 7500 nM T19244 C8SFZ5 70693563 Ki = 60000 nM T19244 C8G4AV 70694560 IC50 > 100000 nM T19244 CC6GZ9 70695067 IC50 > 20000 nM T19244 C75YPE 70695115 IC50 >= 5000 nM T19244 CS1MU4 70695116 IC50 = 9500 nM T19244 C6K9BL 70695117 IC50 = 4500 nM T19244 C1YZ6K 70695118 IC50 = 7200 nM T19244 C53RQN 70695119 IC50 = 4000 nM T19244 CXJ5V2 70695120 IC50 = 5400 nM T19244 CCR12A 70695121 IC50 > 20000 nM T19244 C0WHL2 70695688 Ki = 64000 nM T19244 CVU08A 70695812 IC50 > 25000 nM T19244 C37YJI 70695889 IC50 = 9900 nM T19244 CT1GF8 70697151 IC50 >= 5000 nM T19244 CSX71G 70697153 IC50 = 17000 nM T19244 C4JY5R 70697154 IC50 = 4400 nM T19244 CT78JN 70697155 IC50 > 20000 nM T19244 C34WHG 70697225 IC50 = 3162.28 nM T19244 CJ2GV4 70697669 Ki = 93000 nM T19244 CBDL19 70792359 IC50 > 100000 nM T19244 C7DO1N 70817239 IC50 > 20000 nM T19244 C6L7FH 70817382 IC50 = 5000 nM T19244 C2PJ1D 70865101 IC50 > 30000 nM T19244 C2TC8W 70914230 IC50 > 100000 nM T19244 CXW7U0 70977933 IC50 > 10000 nM T19244 C1VMF2 70977969 IC50 > 50000 nM T19244 CA6GI0 70993878 IC50 = 8100 nM T19244 CK0BD4 71009508 IC50 = 250 nM T19244 C1DUO9 71009649 IC50 = 800 nM T19244 C2HGI7 71153408 IC50 > 10000 nM T19244 C62ULC 71225056 IC50 > 100000 nM T19244 C7Y2LB 71230234 IC50 > 10000 nM T19244 C5RE4T 71244643 IC50 > 10000 nM T19244 C9AT8D 71263621 IC50 = 2600 nM T19244 C6BE5X 71271461 IC50 > 50000 nM T19244 C5L8SW 71279563 IC50 = 4000 nM T19244 CV96FO 71279672 IC50 = 8000 nM T19244 C6RHS3 71279723 IC50 > 8000 nM T19244 CZY5P7 71279859 IC50 = 5000 nM T19244 CGI01S 71280152 IC50 = 4000 nM T19244 C7PLS6 71285927 IC50 = 2100 nM T19244 CAO07V 71293843 IC50 = 500 nM T19244 CWN2M1 71300316 IC50 = 3000 nM T19244 C03KNO 71300317 IC50 = 3100 nM T19244 CWY4S0 71304814 IC50 = 7200 nM T19244 CS9OV5 71315139 IC50 > 100000 nM T19244 C4CT6B 71374169 Ki = 29000 nM T19244 CR37DA 71419478 IC50 = 19952.62 nM T19244 C5SML3 71449452 IC50 = 19952.62 nM T19244 CL6BC1 71449606 IC50 = 4500 nM T19244 C5Q2NY 71452771 Ki = 14000 nM T19244 CZ7GW9 71452855 IC50 = 10 nM T19244 COQ0P1 71453071 IC50 = 19952.62 nM T19244 CSL01M 71454248 IC50 = 1258.93 nM T19244 C47GYB 71454279 IC50 > 10000 nM T19244 CR18YP 71454541 Ki = 7000 nM T19244 C0YD9K 71455398 IC50 = 3000 nM T19244 C4O2GZ 71457203 IC50 = 22400 nM T19244 CF5XH0 71458127 Ki = 21000 nM T19244 C8Q3LC 71460007 Ki = 100 nM T19244 C9DEM5 71461693 Ki = 13000 nM T19244 CL4EO3 71461720 Ki = 25000 nM T19244 CD81EJ 71463058 IC50 = 9100 nM T19244 C0GBL7 71466345 IC50 > 20000 nM T19244 CV78KN 71471711 IC50 = 76850 nM T19244 CFA9V1 71494937 IC50 = 22000 nM T19244 C8U0TA 71510812 IC50 > 25000 nM T19244 C9DIK2 71512060 IC50 > 10000 nM T19244 CF05BU 71513157 IC50 > 10000 nM T19244 CS1ZX0 71513822 IC50 > 10000 nM T19244 C0VLE3 71516457 IC50 = 3500 nM T19244 C2LVY0 71516458 IC50 = 8200 nM T19244 CA07TC 71517197 IC50 > 10000 nM T19244 C3CT1R 71530223 IC50 > 10000 nM T19244 CN8CM1 71533722 IC50 = 21000 nM T19244 C67ZSQ 71540073 IC50 > 30000 nM T19244 C3RQP5 71542927 IC50 = 3100 nM T19244 C1GUX2 71542931 IC50 = 6100 nM T19244 C0IK7U 71544354 IC50 = 9.2 nM T19244 C9N7YA 71544706 IC50 = 1600 nM T19244 C92NEY 71544707 IC50 = 19000 nM T19244 C83YJF 71544946 IC50 > 50000 nM T19244 C4N3OC 71545856 IC50 = 6700 nM T19244 CCN01X 71547862 IC50 > 10000 nM T19244 CKB12X 71549359 IC50 = 19000 nM T19244 C4LZM6 71549637 IC50 = 8000 nM T19244 C6JOB5 71549767 IC50 = 40000 nM T19244 CV47CJ 71549769 IC50 = 13000 nM T19244 C5IV9D 71549913 IC50 = 18000 nM T19244 CSHT69 71550657 IC50 > 19000 nM T19244 C9P5KT 71556166 IC50 > 50000 nM T19244 C8JOU5 71556223 IC50 > 50000 nM T19244 C25XGY 71556353 IC50 = 21000 nM T19244 CP0J5L 71556425 IC50 = 13000 nM T19244 CB5QR3 71556493 IC50 = 12000 nM T19244 CIXL34 71556883 IC50 = 11000 nM T19244 CZ3A7E 71556887 IC50 = 9700 nM T19244 CY59CA 71557630 IC50 = 630 nM T19244 CTI52S 71557789 IC50 = 880 nM T19244 CMKH30 71558122 IC50 > 10000 nM T19244 CS8M1O 71558621 IC50 = 570 nM T19244 CJXK67 71559365 IC50 = 170 nM T19244 C30ZKJ 71561420 IC50 > 100000 nM T19244 CLR92N 71579539 IC50 = 31200 nM T19244 C84GAB 71580631 IC50 > 100000 nM T19244 C4S1TN 71580827 IC50 = 50500 nM T19244 C6CHY1 71580912 IC50 = 9100 nM T19244 CUJT21 71582799 IC50 > 10000 nM T19244 CWD2Z5 71585566 IC50 > 10000 nM T19244 CCE7T2 71585568 IC50 > 10000 nM T19244 C4GNJ3 71598545 IC50 > 10000 nM T19244 C1M7JD 71599971 IC50 > 40000 nM T19244 C0WAH3 71602807 IC50 = 1100 nM T19244 C9J0EH 71603917 IC50 > 50000 nM T19244 CI4PG7 71607631 IC50 = 8820 nM T19244 CKPV51 71621803 IC50 = 138000 nM T19244 C8SGK6 71624246 IC50 = 5000 nM T19244 C2WJX0 71626755 IC50 > 50000 nM T19244 C26TXG 71626895 IC50 > 50000 nM T19244 C4DHC9 71626896 IC50 > 50000 nM T19244 CX0VE7 71626971 IC50 > 50000 nM T19244 C7KJN8 71654714 IC50 = 74 nM T19244 CYD9P8 71654715 IC50 = 515 nM T19244 CWZ83T 71654716 IC50 = 460 nM T19244 CB7H3S 71654717 IC50 = 149 nM T19244 CRM61V 71654718 IC50 > 10000 nM T19244 C3W2YJ 71654788 IC50 = 601 nM T19244 CU50AM 71654790 IC50 = 554 nM T19244 CSV81U 71654791 IC50 = 1140 nM T19244 CT34VN 71654792 IC50 > 10000 nM T19244 C4BMW8 71654793 IC50 > 10000 nM T19244 CCH0T6 71654852 IC50 > 10000 nM T19244 CVEW58 71654853 IC50 > 10000 nM T19244 C8WT4B 71654854 IC50 > 10000 nM T19244 C6QT9L 71654855 IC50 = 2180 nM T19244 C4CB5Y 71654856 IC50 = 930 nM T19244 CG1W6H 71654857 IC50 = 110 nM T19244 C43EHA 71654926 IC50 > 10000 nM T19244 C6I3VF 71654927 IC50 > 10000 nM T19244 CO6K8D 71654928 IC50 > 10000 nM T19244 C8UVZ0 71654929 IC50 > 10000 nM T19244 CJYU32 71654930 IC50 > 10000 nM T19244 CCUW57 71655311 IC50 > 25000 nM T19244 CN13KW 71655312 IC50 > 25000 nM T19244 CHR1L4 71655313 IC50 = 11000 nM T19244 CHZ0U6 71655314 IC50 = 2000 nM T19244 CXT60O 71655374 IC50 > 25000 nM T19244 C9AIJ7 71655375 IC50 > 25000 nM T19244 CGLA96 71655376 IC50 > 25000 nM T19244 C8OX4Q 71655377 IC50 > 25000 nM T19244 C49YGB 71655378 IC50 > 25000 nM T19244 CH7KA2 71655379 IC50 > 25000 nM T19244 C39HIB 71655380 IC50 > 25000 nM T19244 CG9P3O 71655442 IC50 = 63 nM T19244 CXW48Z 71655443 IC50 = 10000 nM T19244 CM2P0R 71655444 IC50 = 400 nM T19244 CSP95X 71655445 IC50 = 400 nM T19244 C2PL3H 71655503 IC50 = 1800 nM T19244 C1FNK2 71655701 IC50 = 4600 nM T19244 CIA03F 71655702 IC50 > 10000 nM T19244 CF68KU 71655703 IC50 > 10000 nM T19244 CQ1NY6 71655704 IC50 > 10000 nM T19244 CFU86J 71655705 IC50 = 125 nM T19244 CDO29V 71655706 IC50 = 644 nM T19244 CDL35U 71655748 IC50 > 5000 nM T19244 CG4HW8 71655768 IC50 = 1960 nM T19244 CL56VA 71655769 IC50 > 10000 nM T19244 CS2EN8 71655770 IC50 = 139 nM T19244 C6VRC0 71655771 IC50 = 1300 nM T19244 C7UA4I 71655772 IC50 > 10000 nM T19244 CPB6T3 71655773 IC50 = 1770 nM T19244 CAN6X5 71656574 IC50 = 16000 nM T19244 C61RYH 71659356 IC50 > 30000 nM T19244 CVDB58 71659357 IC50 > 30000 nM T19244 C28EIT 71659358 IC50 > 30000 nM T19244 C8DF4B 71659489 IC50 > 30000 nM T19244 C7Y0RM 71659490 IC50 > 30000 nM T19244 CKR47S 71659491 IC50 = 21000 nM T19244 CAQ2V1 71659492 IC50 > 30000 nM T19244 CJX32Y 71659493 IC50 > 30000 nM T19244 C05JLG 71659494 IC50 > 30000 nM T19244 COS6Q5 71659610 IC50 = 5200 nM T19244 CNVI07 71659611 IC50 > 30000 nM T19244 CUF06Z 71659612 IC50 > 30000 nM T19244 CT9KZ0 71659613 IC50 > 30000 nM T19244 CZFU74 71659614 IC50 > 30000 nM T19244 CC3L1Y 71659615 IC50 > 30000 nM T19244 CF1HA9 71659751 IC50 = 25000 nM T19244 CF8DV2 71659752 IC50 > 30000 nM T19244 CMA4N0 71659753 IC50 = 17000 nM T19244 CFBA41 71659754 IC50 = 9000 nM T19244 CR58TZ 71659755 IC50 > 30000 nM T19244 CVE91N 71659756 IC50 = 21000 nM T19244 CH4VF0 71659894 IC50 > 30000 nM T19244 C53AOG 71659895 IC50 > 30000 nM T19244 C9WC2J 71659896 IC50 > 30000 nM T19244 CTBX46 71659897 IC50 = 9800 nM T19244 CW0Y5N 71659898 IC50 = 20000 nM T19244 CZD71P 71680760 IC50 > 30000 nM T19244 CY8VM4 71695585 IC50 > 10000 nM T19244 C8LE5D 71695973 IC50 > 10000 nM T19244 CMAW93 71711804 IC50 > 10000 nM T19244 C9I3GO 71714121 IC50 > 50000 nM T19244 CO6Q3R 71715127 IC50 > 10000 nM T19244 C6JS5H 71715183 IC50 = 7200 nM T19244 CYR2J8 71715184 IC50 > 10000 nM T19244 C6JS5R 71715185 IC50 > 10000 nM T19244 CHS3X9 71715186 IC50 > 10000 nM T19244 CIX79H 71715241 IC50 > 10000 nM T19244 CC4A3K 71716821 IC50 = 321 nM T19244 CUG2V3 71716866 IC50 = 517 nM T19244 CIZ40M 71716873 IC50 = 3234 nM T19244 C4XYN9 71717494 IC50 = 1365 nM T19244 C89GSF 71718127 IC50 = 1012 nM T19244 CWB3V1 71718136 IC50 = 13300 nM T19244 C7TM8H 71718630 IC50 = 1368 nM T19244 CW38FM 71718726 IC50 = 39 nM T19244 CY6D2J 71719903 IC50 = 37 nM T19244 CL0O5N 71719912 IC50 = 205 nM T19244 CYQH30 71719914 IC50 = 100 nM T19244 C1FYA8 71720426 IC50 > 20000 nM T19244 CMDI34 71720470 IC50 = 180 nM T19244 C7B8UH 71720543 IC50 = 279 nM T19244 CQEH46 71720911 IC50 = 720 nM T19244 C30NBJ 71722055 IC50 > 10000 nM T19244 CIN10C 71727133 IC50 > 10000 nM T19244 CB53IQ 71727461 IC50 = 77 nM T19244 C2SQ6K 71727682 IC50 = 80 nM T19244 CLE15B 71727801 IC50 = 70 nM T19244 CV6QC1 71727805 IC50 > 10000 nM T19244 CE8R1D 71727929 IC50 = 3900 nM T19244 C6USH8 71727930 IC50 = 73 nM T19244 C1W4DX 71727932 IC50 = 65 nM T19244 C36DNH 71727934 IC50 > 10000 nM T19244 CJZR51 71728054 IC50 = 200 nM T19244 CQ21ZD 71733911 IC50 > 50000 nM T19244 C56MYK 71739468 IC50 > 30000 nM T19244 C60BIX 71763463 IC50 = 40 nM T19244 CJHI28 71770158 IC50 = 2430 nM T19244 C9LU5Q 71770282 IC50 = 3140 nM T19244 CTSK68 71811225 IC50 = 9100 nM T19244 CVL54T 71811261 IC50 = 2100 nM T19244 CH8M5Y 71811363 IC50 > 50000 nM T19244 C1WT8V 71811365 IC50 > 50000 nM T19244 C5JV1P 71812623 EC50 > 100000 nM T19244 CJH9K3 71814859 IC50 > 10000 nM T19244 CD28XR 71816087 IC50 > 10000 nM T19244 CC4SU1 71817351 IC50 = 300 nM T19244 CY04LE 71817500 IC50 = 270 nM T19244 C6EC3O 72163432 IC50 > 30000 nM T19244 CNF81W 72163837 IC50 > 30000 nM T19244 CB2NP7 72165228 IC50 > 20000 nM T19244 C2OV4Z 72189207 IC50 > 10000 nM T19244 CW4E9O 72189514 IC50 = 800 nM T19244 CAVB46 72189515 IC50 = 6900 nM T19244 C4KUM3 72189516 IC50 > 10000 nM T19244 CR5Y6U 72189517 IC50 > 10000 nM T19244 C46FSX 72189518 IC50 > 10000 nM T19244 CBW0G9 72189519 IC50 > 10000 nM T19244 CC0DB5 72189807 IC50 > 10000 nM T19244 CUQ69N 72189808 IC50 > 10000 nM T19244 C1V7PU 72189809 IC50 > 10000 nM T19244 CC1SR3 72189810 IC50 > 10000 nM T19244 C9NCE7 72189811 IC50 > 10000 nM T19244 C2ZF9X 72190130 IC50 > 10000 nM T19244 CXH2S6 72190131 IC50 > 10000 nM T19244 C12KEZ 72190132 IC50 > 10000 nM T19244 CW64OR 72190133 IC50 > 10000 nM T19244 CWT7K2 72205601 IC50 = 8910 nM T19244 CE46KA 72375120 IC50 > 30000 nM T19244 CHVL93 72375121 IC50 > 30000 nM T19244 CK7DE4 72545105 IC50 > 20000 nM T19244 C4G2UR 72695027 IC50 > 10000 nM T19244 CDFO42 72695136 IC50 > 10000 nM T19244 CK7F6U 72700776 IC50 > 10000 nM T19244 CM75FY 72703989 IC50 > 25000 nM T19244 CPQ34Z 72703991 IC50 > 25000 nM T19244 CBE48L 72707143 IC50 > 10000 nM T19244 C9OQ2I 72710839 IC50 = 900 nM T19244 C7A5EW 72714054 IC50 > 50000 nM T19244 C7SZ3V 72714058 IC50 > 50000 nM T19244 C3J0ZB 72725671 IC50 = 10300 nM T19244 C8QEJ3 72725792 IC50 > 50000 nM T19244 C7AO4X 72792633 IC50 > 50000 nM T19244 CLK7O4 72792692 IC50 > 50000 nM T19244 CBM7W0 72793032 IC50 = 1900 nM T19244 CNHI43 72793033 IC50 = 2900 nM T19244 C5E7IF 72793034 IC50 = 4900 nM T19244 CR4U6G 72793098 IC50 = 5000 nM T19244 CX38EH 72793099 IC50 > 40000 nM T19244 CNFA68 72793323 IC50 = 14000 nM T19244 CHW6N1 72793324 IC50 > 40000 nM T19244 C8G0MY 72793393 IC50 > 40000 nM T19244 C6R8DI 72943374 IC50 > 20000 nM T19244 C59QLH 72943630 IC50 = 1380 nM T19244 C9WU2M 72950813 IC50 > 100000 nM T19244 C1QMY5 73053248 IC50 > 10000 nM T19244 CH1JK9 73213123 IC50 > 40000 nM T19244 C7B2VH 73332466 IC50 = 7900 nM T19244 C57LGA 73349098 IC50 > 10000 nM T19244 C80BSO 73352560 IC50 > 20000 nM T19244 CG7R3F 73353420 IC50 > 30000 nM T19244 CM0W7S 73354069 IC50 > 20000 nM T19244 CRA5H6 73389570 IC50 > 10000 nM T19244 CDX9R1 73603344 IC50 > 50000 nM T19244 CTMF86 73603391 IC50 > 50000 nM T19244 C7LER5 73669500 IC50 > 50000 nM T19244 CJKB83 73670174 IC50 > 50000 nM T19244 CHV3W1 73774630 IC50 > 30000 nM T19244 CYV4Z6 73890929 IC50 = 340 nM T19244 CCFI76 73890932 IC50 = 1000 nM T19244 C15QVF 74221424 IC50 > 100000 nM T19244 CZ3TB5 74221949 IC50 > 50000 nM T19244 CW9N8T 74222036 IC50 > 50000 nM T19244 CUF63H 74223858 IC50 = 3000 nM T19244 COE76R 74223859 IC50 = 31 nM T19244 C7RAQ4 74538704 IC50 > 20000 nM T19244 CPS18J 75276948 EC50 = 7000 nM T19244 C2G8VR 75593287 IC50 > 25000 nM T19244 C9E0PX 76071764 IC50 = 780 nM T19244 C1Y7HC 76072411 IC50 = 1500 nM T19244 C20YHA 76283431 IC50 > 30000 nM T19244 CHV72I 76283681 IC50 > 20000 nM T19244 CT59ZA 76283684 IC50 > 20000 nM T19244 CE2NP9 76284760 IC50 > 20000 nM T19244 C7ZM6V 76310313 IC50 > 100000 nM T19244 C7JAY2 76310561 IC50 = 3400 nM T19244 CQY40K 76310562 IC50 > 25000 nM T19244 CA70YQ 76310589 IC50 > 30000 nM T19244 CY0HD7 76311092 IC50 = 570 nM T19244 CAT65E 76311096 IC50 = 490 nM T19244 CF07EK 76313382 IC50 > 20000 nM T19244 CQFG10 76314530 IC50 > 50000 nM T19244 CX3LZ0 76314702 IC50 = 450 nM T19244 CJO15N 76316894 IC50 > 20000 nM T19244 C3OP2B 76319044 IC50 > 10000 nM T19244 CEK3O5 76321713 IC50 > 30000 nM T19244 CNY2D6 76321910 EC50 > 40000 nM T19244 C7Y5QF 76321979 IC50 = 900 nM T19244 CR05PL 76322043 IC50 > 100000 nM T19244 CQ3CW1 76322044 IC50 = 67200 nM T19244 CYXU43 76322162 IC50 > 30000 nM T19244 C2SM8Y 76325108 IC50 > 30000 nM T19244 C1HJQ9 76325597 IC50 = 910 nM T19244 CYR3L4 76327922 IC50 > 50000 nM T19244 CJ9N0S 76328675 IC50 > 30000 nM T19244 C5UMK8 76328829 IC50 > 30000 nM T19244 C8CQ9Y 76328873 IC50 > 30000 nM T19244 CZ9Q2S 76329164 IC50 > 10000 nM T19244 CWD5R4 76331595 IC50 > 50000 nM T19244 CZ2CQ7 76332826 IC50 = 7800 nM T19244 C76UKL 76333454 IC50 > 20000 nM T19244 C9QYB2 76335964 IC50 = 13800 nM T19244 CE4YP9 76335969 IC50 > 10000 nM T19244 CGE5S3 76336366 EC50 > 40000 nM T19244 CGJM01 76336447 IC50 > 10000 nM T19244 C92WBQ 76336500 IC50 > 100000 nM T19244 C10CNR 76684033 IC50 < 10000 nM T19244 CAT95V 76685067 IC50 = 43230 nM T19244 C7F2RD 77050711 IC50 = 99000 nM T19244 CRI9Z8 77107273 IC50 = 5200 nM T19244 CWG4T2 78209992 IC50 > 50 nM T19244 CLB1A4 78319901 IC50 > 50000 nM T19244 C9GQS2 81689815 IC50 = 82000 nM T19244 C3H5XR 82639722 IC50 > 10000 nM T19244 CQMB31 85470872 IC50 > 10000 nM T19244 C15BSO 86270136 IC50 > 10000 nM T19244 CA1CE3 86270720 IC50 > 10000 nM T19244 C9TE7X 86271008 IC50 > 10000 nM T19244 CMZV56 86271009 IC50 > 10000 nM T19244 CXN93A 86271108 IC50 > 10000 nM T19244 C2KHM0 86271111 IC50 > 10000 nM T19244 CZL23E 86271138 IC50 = 2000 nM T19244 C5IR2K 86271238 IC50 > 30000 nM T19244 CN9MO7 86271494 IC50 > 10000 nM T19244 C4T3IW 86272102 IC50 = 45000 nM T19244 C13AJC 86274362 IC50 = 56000 nM T19244 C3OLB1 86274489 IC50 = 7000 nM T19244 CAB78T 86274732 IC50 = 77000 nM T19244 CCU13T 86275207 IC50 = 12000 nM T19244 CJ68CO 86275449 IC50 = 42000 nM T19244 CF4QX9 86278359 IC50 > 10000 nM T19244 CXF9Q3 86279146 IC50 > 30000 nM T19244 C4Y3VP 86279147 IC50 > 30000 nM T19244 CH3FN8 86288905 IC50 = 19000 nM T19244 CKQ71X 86288935 IC50 = 5350 nM T19244 C36LAF 86302354 IC50 > 25000 nM T19244 C98BAP 86302469 IC50 = 19000 nM T19244 C6A1DG 86304283 IC50 = 5600 nM T19244 C0IZU4 86304284 IC50 = 13000 nM T19244 C5JFM1 86304285 IC50 = 330 nM T19244 CKJI10 86304439 IC50 = 580 nM T19244 CGK31H 86304440 IC50 = 8700 nM T19244 CJ7SI6 86304441 IC50 = 27000 nM T19244 C9EMQ0 86304601 IC50 > 34000 nM T19244 CV4Q5D 86304762 IC50 = 17000 nM T19244 CK02ZT 86344136 IC50 = 4700 nM T19244 CZU43C 86344330 IC50 = 1200 nM T19244 C6D5QL 86344510 IC50 = 13000 nM T19244 CM3AE5 86344511 IC50 = 17000 nM T19244 C1UZ7Y 86344512 IC50 = 6100 nM T19244 CJC7V3 86344877 IC50 = 2800 nM T19244 C3SIV1 86345235 IC50 = 78 nM T19244 CMXZ65 86346192 IC50 > 10000 nM T19244 CG7T0R 86582124 IC50 = 100 nM T19244 CMG39E 86673884 IC50 > 20000 nM T19244 CVJ8L5 86728666 IC50 = 3300 nM T19244 CQ45XR 86763358 IC50 > 15848.93 nM T19244 CTW8L6 86766622 IC50 = 5200 nM T19244 C2U0BG 87055263 IC50 = 3200 nM T19244 CF67AV 88875879 IC50 > 100000 nM T19244 CL7NM6 89452242 IC50 = 1000 nM T19244 CR0EY3 89452445 IC50 = 1000 nM T19244 C8Y9RW 89462922 IC50 = 3.4 nM T19244 C0DRH8 89463724 IC50 = 2.7 nM T19244 C8SK1N 89463725 IC50 = 6.5 nM T19244 CL30TR 89471870 IC50 > 25000 nM T19244 CA49UY 89726151 IC50 > 30000 nM T19244 CY6K5P 89738540 IC50 > 30000 nM T19244 CIXB02 89738547 IC50 > 30000 nM T19244 CG9CM0 89750383 IC50 = 6900 nM T19244 COU52N 89761779 IC50 = 250 nM T19244 C2BM9L 89768534 IC50 > 30000 nM T19244 CB4Y7R 89768546 IC50 > 30000 nM T19244 C5MR9K 89777151 IC50 > 30000 nM T19244 CRZ34V 89777258 IC50 = 2300 nM T19244 CZ58KT 89777437 IC50 = 26000 nM T19244 C5S4PX 89777463 IC50 = 25000 nM T19244 C9I6NQ 89789762 IC50 = 9400 nM T19244 C1QDJ0 89793388 IC50 > 10000 nM T19244 CUS70D 89793496 IC50 = 1000 nM T19244 CP7MZ2 89793516 IC50 = 160 nM T19244 C9X5OT 89793519 IC50 = 70 nM T19244 C96EWN 89795484 IC50 = 300 nM T19244 CWO58S 89795501 IC50 = 200 nM T19244 CIQ53M 89795553 IC50 = 1900 nM T19244 C5GQL0 89795796 IC50 = 190 nM T19244 C16AXO 89846366 IC50 > 50000 nM T19244 CEK2I7 89846957 IC50 > 20000 nM T19244 C4MJ6O 89846958 IC50 > 50000 nM T19244 CMS6X4 89931025 IC50 > 20000 nM T19244 CQ5HZ7 89996234 IC50 > 50000 nM T19244 CJ65EF 90012001 IC50 > 10000 nM T19244 C6KYB4 90012693 IC50 > 10000 nM T19244 CG78UF 90013202 IC50 > 10000 nM T19244 CIOZ97 90013255 IC50 > 10000 nM T19244 C3YPA8 90149424 IC50 = 2100 nM T19244 C1Q6PT 90149477 IC50 = 7300 nM T19244 CY5IC7 90252834 IC50 = 9100 nM T19244 C84NVA 90252850 IC50 = 11000 nM T19244 CBY46O 90252851 IC50 = 7200 nM T19244 CNVA50 90252852 IC50 = 3800 nM T19244 CRN8G1 90253396 IC50 > 20000 nM T19244 CFG74P 90408756 IC50 = 5500 nM T19244 CE4IT5 90408860 IC50 > 10000 nM T19244 CJPC93 90410264 IC50 = 1200 nM T19244 C2FKB3 90410598 IC50 = 1600 nM T19244 CB0RP3 90410604 IC50 = 2800 nM T19244 CQ8ZW3 90410911 IC50 > 10000 nM T19244 CD5W6K 90417914 IC50 = 14000 nM T19244 C1EVN3 90455889 IC50 = 2500 nM T19244 CAGK52 90456097 IC50 = 3700 nM T19244 CJE7P5 90467013 IC50 > 50000 nM T19244 CX6DQ4 90467014 IC50 > 50000 nM T19244 C7D2UK 90467156 IC50 > 50000 nM T19244 CV75ZC 90467159 IC50 > 50000 nM T19244 C3RO1M 90467162 IC50 > 50000 nM T19244 CF30KA 90643570 IC50 > 100000 nM T19244 CGS36U 90644505 IC50 > 25000 nM T19244 CYE3G5 90644506 IC50 > 25000 nM T19244 CDE57X 90644507 IC50 > 25000 nM T19244 CV53YI 90644508 IC50 > 10000 nM T19244 C9FCS1 90644592 IC50 = 14000 nM T19244 C1S8PM 90644647 IC50 > 30000 nM T19244 C5WDB0 90644648 IC50 > 30000 nM T19244 C5O8HN 90644762 IC50 = 27900 nM T19244 CY4PB3 90644766 IC50 > 30000 nM T19244 CL5UB3 90644769 IC50 = 22900 nM T19244 C6AMK9 90644770 IC50 > 30000 nM T19244 CAVN86 90644773 IC50 > 30000 nM T19244 CEZK64 90645309 IC50 > 20000 nM T19244 CXUH46 90645310 IC50 > 20000 nM T19244 C0NM1C 90645311 IC50 = 1900 nM T19244 CL0O7Q 90645312 IC50 > 20000 nM T19244 CHP74S 90654587 IC50 = 4700 nM T19244 C96YCU 90654600 IC50 > 25000 nM T19244 CIL2W9 90664452 IC50 = 3300 nM T19244 CSDO81 90664458 IC50 > 25000 nM T19244 CQT69X 90664721 IC50 > 100000 nM T19244 CN3A1P 90664848 IC50 > 100000 nM T19244 CJ01LW 90664969 IC50 > 100000 nM T19244 CG98QO 90665194 IC50 = 2900 nM T19244 C02PLA 90665208 IC50 > 100000 nM T19244 CXEJ32 90665986 IC50 > 30000 nM T19244 CDQ56W 90665987 IC50 > 30000 nM T19244 C5E2FJ 90665988 IC50 > 30000 nM T19244 CXEK45 90681222 IC50 > 30000 nM T19244 C8H4KE 90681223 IC50 > 30000 nM T19244 CA9PL8 91663316 IC50 = 8200 nM T19244 C65ANP 91666625 IC50 > 40000 nM T19244 C26BZK 91666633 IC50 > 10000 nM T19244 C9ETC1 91666645 IC50 > 50000 nM T19244 C2H7XV 91668260 IC50 > 5000 nM T19244 C4YP6M 91754658 IC50 = 25000 nM T19244 C5CKD3 91754690 IC50 > 20000 nM T19244 CM95VC 91758806 IC50 = 1290 nM T19244 C5T0FH 91799687 IC50 > 10000 nM T19244 CUX4B6 91809187 IC50 > 60000 nM T19244 CUQ1W0 91810395 IC50 = 15700 nM T19244 CWTO83 91810751 IC50 > 10000 nM T19244 CC9B6T 91820646 IC50 > 18000 nM T19244 C3L6KU 91820689 IC50 > 25000 nM T19244 CL7S4U 91844670 IC50 > 10000 nM T19244 C1JPD6 91844700 IC50 > 10000 nM T19244 CSK6Z1 91844707 IC50 = 5900 nM T19244 CH4L7O 91885483 IC50 > 30000 nM T19244 CBG6E7 91885506 IC50 > 5600 nM T19244 CF8W2B 91928421 IC50 = 2900 nM T19244 CU1G3S 91933941 IC50 > 10000 nM T19244 CWZX73 91971958 IC50 = 3500 nM T19244 C57QJY 92045044 EC50 = 277 nM T19244 C38ZID 92045057 IC50 > 10000 nM T19244 CM6VG1 92239323 IC50 > 20000 nM T19244 CY2UI5 101891769 IC50 > 30000 nM T19244 CGB54P 101902999 IC50 = 900 nM T19244 CG62HP 101903000 IC50 = 2500 nM T19244 C87GEW 102435977 IC50 > 10000 nM T19244 CQ9PN8 102593934 IC50 = 14500 nM T19244 C4Z1OU 110451319 IC50 = 10000 nM T19244 CN57AX 110451673 IC50 = 10000 nM T19244 CYX7T2 117072549 IC50 > 50000 nM T19244 C8F6VO 117604931 IC50 = 42000 nM T19244 CNFW42 117608566 IC50 > 10000 nM T19244 CGL3R6 117614609 IC50 = 1000 nM T19244 C6O7ZX 117736868 IC50 = 4000 nM T19244 CV94EU 117736992 IC50 = 560 nM T19244 CVI38D 117737118 IC50 = 2900 nM T19244 CI0D1R 117737120 IC50 = 2300 nM T19244 C23NPF 117737172 IC50 = 8200 nM T19244 CM1T3I 117737215 IC50 = 2600 nM T19244 CN1E5U 117737262 IC50 = 580 nM T19244 CS4IW2 117739617 IC50 = 1900 nM T19244 CFJ97D 117741583 IC50 = 1900 nM T19244 CUZ6C2 117741590 IC50 = 4200 nM T19244 C0V3KH 117741592 IC50 = 1300 nM T19244 CBL12U 117748926 IC50 = 2100 nM T19244 C10BKY 117749324 IC50 = 4600 nM T19244 CS72RV 117885758 IC50 > 50000 nM T19244 C6Z3NJ 117885766 IC50 > 50000 nM T19244 CKU6S4 117885912 IC50 > 50000 nM T19244 C89EQN 117897570 IC50 > 7200 nM T19244 C9KV7L 117993993 IC50 = 45300 nM T19244 CNV24M 117993998 IC50 = 34100 nM T19244 CGBO72 118016229 IC50 > 20000 nM T19244 CJB47R 118086034 IC50 = 13000 nM T19244 C3TBD8 118103460 IC50 > 30000 nM T19244 CZR2Q1 118103881 IC50 = 1600 nM T19244 CL15XC 118103886 IC50 = 1000 nM T19244 CI9Q2H 118103892 IC50 = 5700 nM T19244 CI3KM2 118103909 IC50 > 30000 nM T19244 CAIU03 118104096 IC50 = 20500 nM T19244 CIL65X 118104099 IC50 = 6900 nM T19244 CMX3U8 118107483 IC50 >= 5000 nM T19244 CWR6I1 118112300 IC50 > 20000 nM T19244 CNM1W9 118141977 IC50 = 8010 nM T19244 C56INY 118142016 IC50 = 5900 nM T19244 CN1LC9 118142017 IC50 = 6400 nM T19244 CZ0E5W 118142030 IC50 = 16000 nM T19244 CW5N0O 118142047 IC50 = 3800 nM T19244 CR4DE7 118175009 IC50 > 10000 nM T19244 CO9P5Y 118207089 IC50 = 4300 nM T19244 C2U3TJ 118208018 IC50 > 20000 nM T19244 C6HSC3 118217854 IC50 > 10000 nM T19244 CEKH57 118217858 IC50 > 10000 nM T19244 CRM37Z 118223719 IC50 = 3400 nM T19244 CEN18L 118224069 IC50 = 17600 nM T19244 CT42ZR 118261815 IC50 > 50000 nM T19244 C3R9TY 118324047 IC50 > 10000 nM T19244 C7AO1M 118324066 IC50 > 10000 nM T19244 CPO08K 118344339 IC50 = 8600 nM T19244 CTCQ02 118344344 IC50 = 9500 nM T19244 C1HX3A 118344346 IC50 > 20000 nM T19244 CI7P6J 118344348 IC50 > 20000 nM T19244 C8J1PY 118344351 IC50 > 20000 nM T19244 CAWZ16 118344383 IC50 > 20000 nM T19244 CSUK24 118344385 IC50 > 20000 nM T19244 CA1YM6 118344504 IC50 = 2700 nM T19244 CC3N6Z 118344616 IC50 = 10000 nM T19244 CC0RD7 118345442 IC50 > 20000 nM T19244 CK43EA 118345549 IC50 = 13000 nM T19244 C0MCW3 118346170 IC50 > 20000 nM T19244 CRZ5N1 118368912 IC50 > 50000 nM T19244 CBIR89 118389918 IC50 = 22700 nM T19244 CR7DJ0 118453722 IC50 > 50000 nM T19244 CK1Z7I 118462026 IC50 > 50000 nM T19244 CM2NH5 118478848 IC50 = 23400 nM T19244 CRV8S3 118478927 IC50 > 10000 nM T19244 CL32JE 118478933 IC50 > 10000 nM T19244 C5S1HZ 118478972 IC50 > 10000 nM T19244 C8G9HP 118478986 IC50 > 10000 nM T19244 CBV89G 118478994 IC50 > 10000 nM T19244 CK0ER5 118478999 IC50 > 10000 nM T19244 CU25KC 118479000 IC50 > 10000 nM T19244 CW07IS 118479006 IC50 > 10000 nM T19244 C3ZAV0 118479034 IC50 > 10000 nM T19244 C4W6ZS 118479038 IC50 > 10000 nM T19244 CRG24C 118479053 IC50 > 10000 nM T19244 CD4ME1 118479123 IC50 > 10000 nM T19244 CB0XM2 118479161 IC50 > 10000 nM T19244 C18NTQ 118479199 IC50 > 10000 nM T19244 CJ0Z1Y 118479222 IC50 > 10000 nM T19244 CP0U6Y 118479229 IC50 > 10000 nM T19244 C3A6HD 118479231 IC50 > 10000 nM T19244 CJ14CR 118479241 IC50 > 10000 nM T19244 C1FO3N 118479293 IC50 > 10000 nM T19244 CF02TZ 118479295 IC50 > 10000 nM T19244 C90TED 118479305 IC50 > 10000 nM T19244 C7I9RC 118479316 IC50 > 10000 nM T19244 CRC4F6 118479354 IC50 > 10000 nM T19244 CRCV51 118479359 IC50 > 10000 nM T19244 CJL5W0 118479428 IC50 > 10000 nM T19244 CS2VA7 118479440 IC50 > 10000 nM T19244 CJ9P0M 118479445 IC50 > 10000 nM T19244 C3U1RB 118479452 IC50 > 10000 nM T19244 CBJ28X 118483320 IC50 = 11000 nM T19244 C8PU5O 118491249 IC50 > 10000 nM T19244 C3KAO6 118491258 IC50 > 20000 nM T19244 CINA28 118492166 IC50 > 20000 nM T19244 CJ9Z0S 118496546 IC50 = 4700 nM T19244 C7AYV5 118540795 IC50 = 3750 nM T19244 CB41MH 118560618 IC50 = 22000 nM T19244 C78LNX 118572065 IC50 > 30000 nM T19244 CFH39Z 118621271 IC50 > 10000 nM T19244 C18SWX 118621276 IC50 > 10000 nM T19244 CR6AF2 118621278 IC50 > 10000 nM T19244 C9A5WK 118621285 IC50 > 10000 nM T19244 C9GCH6 118621295 IC50 > 10000 nM T19244 CZR26D 118621302 IC50 > 10000 nM T19244 CP07JL 118621306 IC50 > 10000 nM T19244 C0WV1H 118621308 IC50 > 10000 nM T19244 CF2Q7C 118621309 IC50 > 10000 nM T19244 C9SY5J 118621333 IC50 > 10000 nM T19244 CXU42D 118621370 IC50 > 10000 nM T19244 C4VNM0 118621378 IC50 > 10000 nM T19244 CXL76C 118621380 IC50 > 10000 nM T19244 C4CSN8 118621388 IC50 > 10000 nM T19244 CSU41F 118621392 IC50 > 10000 nM T19244 CT0W3L 118621401 IC50 > 10000 nM T19244 CHFL73 118621409 IC50 > 10000 nM T19244 CYX1L5 118621411 IC50 > 10000 nM T19244 CK87IQ 118621413 IC50 > 10000 nM T19244 C0XJT5 118626089 IC50 > 100000 nM T19244 CRS34C 118705500 IC50 > 100000 nM T19244 CLUN23 118706414 IC50 > 20000 nM T19244 C2BG1F 118706537 IC50 = 1100 nM T19244 C2WP6X 118706538 IC50 = 2200 nM T19244 CZE4U0 118706539 IC50 = 3100 nM T19244 CX8I0G 118706540 IC50 = 2400 nM T19244 CS4R3B 118707826 IC50 > 30000 nM T19244 CLS7C1 118707978 IC50 = 14000 nM T19244 C9LV0M 118707979 IC50 = 7000 nM T19244 CR8VJ2 118708873 IC50 > 5000 nM T19244 CL2VY5 118708881 IC50 > 5000 nM T19244 CB5F2O 118708929 IC50 > 5000 nM T19244 C8M3JX 118708934 IC50 > 5000 nM T19244 C9W3LI 118708938 IC50 > 5000 nM T19244 CEAK31 118708939 IC50 > 5000 nM T19244 CMX6S5 118709259 IC50 > 20000 nM T19244 CT1J7Y 118709777 IC50 = 1540 nM T19244 CT5Y4F 118711210 IC50 = 5500 nM T19244 CFND64 118711211 IC50 > 50000 nM T19244 C4VAE0 118713757 IC50 = 3130 nM T19244 C84GOU 118713773 IC50 = 12900 nM T19244 C2LY9D 118713799 IC50 = 440 nM T19244 CMO2V7 118713801 IC50 = 32700 nM T19244 C9LKI0 118713803 IC50 = 6890 nM T19244 C2OZ7H 118713805 IC50 = 460 nM T19244 CM4P8X 118713806 IC50 = 3340 nM T19244 C7EXQ9 118713807 IC50 = 360 nM T19244 CUM74B 118716060 IC50 > 10000 nM T19244 CLGD29 118720097 IC50 = 5250 nM T19244 C4LW6I 118720885 IC50 > 40000 nM T19244 C9SF2E 118720891 IC50 > 24000 nM T19244 C8VYR0 118721373 IC50 = 4800 nM T19244 CFL73Q 118724203 IC50 = 7000 nM T19244 C6RXB2 118729222 IC50 > 40000 nM T19244 C9HFE1 118730345 IC50 > 10000 nM T19244 C6HV3B 118730351 IC50 > 10000 nM T19244 C3LZM9 118730352 IC50 > 7000 nM T19244 C6B4XD 118730937 IC50 = 6600 nM T19244 CO81CK 118730940 IC50 > 20000 nM T19244 C27FIO 118730943 IC50 > 20000 nM T19244 CLU74Q 118731287 IC50 = 440 nM T19244 C6OEU2 118733374 IC50 > 50000 nM T19244 C4G3YC 118734875 IC50 > 30000 nM T19244 C9AIE1 118734876 IC50 > 30000 nM T19244 C0SM3L 118735340 IC50 < 5000 nM T19244 CAN90V 118735353 IC50 = 17000 nM T19244 C4XY9I 118735354 IC50 = 5000 nM T19244 C1XL4S 118735355 IC50 = 4000 nM T19244 CB57VC 118737720 IC50 > 50000 nM T19244 C15QMA 118737724 IC50 > 50000 nM T19244 C1MHT0 118737725 IC50 > 50000 nM T19244 C5BOQ1 118753201 Ki > 30000 nM T19244 C87ZPY 118796358 IC50 > 50000 nM T19244 CW8SX7 118796776 IC50 = 4000 nM T19244 CIPQ86 118861736 EC50 = 269 nM T19244 CR71BE 118861737 EC50 = 660 nM T19244 CDSY04 118861738 EC50 = 87.7 nM T19244 C9WBY6 118861778 EC50 = 116 nM T19244 CELZ36 118866105 IC50 = 25000 nM T19244 C14DLY 118872292 IC50 = 4700 nM T19244 CM59EQ 118917669 IC50 = 1100 nM T19244 C6J8YF 118917671 IC50 = 350 nM T19244 C2RBF7 118918048 IC50 = 1500 nM T19244 CC4LA1 118953461 IC50 = 11200 nM T19244 C8L1QI 118959080 IC50 > 5000 nM T19244 C9LR8Z 118965395 IC50 > 100000 nM T19244 C13EIL 118967091 IC50 = 6800 nM T19244 CE3CN6 118971057 IC50 = 6100 nM T19244 C4K3PR 118987036 IC50 > 25000 nM T19244 COS3K9 121304408 IC50 > 5000 nM T19244 C9G3ZJ 121304414 IC50 > 7000 nM T19244 C4RD9Y 121304424 IC50 > 17000 nM T19244 C1PKR0 121304441 IC50 > 3000 nM T19244 CC3MP6 121304452 IC50 > 3000 nM T19244 CW68KD 121304458 IC50 > 50000 nM T19244 CPB58L 121304467 IC50 > 9000 nM T19244 COB2X5 121304477 IC50 > 7000 nM T19244 CZ0BI4 121304484 IC50 > 38000 nM T19244 CW51NQ 121304485 IC50 > 17000 nM T19244 CX1DQ6 121304488 IC50 > 6000 nM T19244 C7NLV2 121304500 IC50 > 10000 nM T19244 CPNV43 121304527 IC50 > 17000 nM T19244 CQ2UM4 121304538 IC50 > 17000 nM T19244 C1AB6P 121304551 IC50 > 17000 nM T19244 CN05ZQ 121304574 IC50 > 17000 nM T19244 CU0M7B 121304590 IC50 > 17000 nM T19244 CX5MO3 121304598 IC50 > 6000 nM T19244 C31AEQ 121304649 IC50 > 17000 nM T19244 C2VTK5 121304654 IC50 > 10000 nM T19244 C6IB0P 121304685 IC50 > 21000 nM T19244 CXC70Q 121304711 IC50 > 7000 nM T19244 C6C9EF 121304827 IC50 = 11405 nM T19244 CU4CW1 121313969 IC50 > 50000 nM T19244 C65ZYO 121332604 IC50 > 3000 nM T19244 C92NOH 121332654 IC50 > 3000 nM T19244 CNBH32 121332727 IC50 > 3000 nM T19244 C9Q2ND 121333973 IC50 = 430 nM T19244 C6TBD2 121345502 IC50 > 50000 nM T19244 C4CPO3 121398401 IC50 > 25000 nM T19244 C59ORZ 121398668 IC50 > 10000 nM T19244 CV9TX1 121399281 IC50 = 24850 nM T19244 C2WD1Q 121407246 IC50 = 19820 nM T19244 C9CV7H 121411850 IC50 > 20000 nM T19244 CU3BI0 121412063 IC50 > 20000 nM T19244 CQZ9W3 121414283 IC50 > 25000 nM T19244 C91PVZ 121428416 IC50 > 10000 nM T19244 C3KNZ5 121439991 IC50 > 50000 nM T19244 CE7H5V 121465028 IC50 = 1830 nM T19244 CV5R4G 121470704 IC50 = 11100 nM T19244 C85HZL 121470706 IC50 = 9900 nM T19244 C09QGL 121470709 IC50 = 16000 nM T19244 C3OL2H 121480641 IC50 = 31970 nM T19244 CD89ZC 121480642 IC50 = 13500 nM T19244 CM8NK7 121499158 IC50 > 10000 nM T19244 CHD26A 121596332 IC50 > 20000 nM T19244 C3RFZ1 121596966 IC50 = 373 nM T19244 CP52DJ 121596967 IC50 = 858 nM T19244 C9WB6E 122179416 IC50 > 100000 nM T19244 CYFA75 122179419 IC50 = 8543 nM T19244 CNGQ19 122179477 IC50 > 10000 nM T19244 C8M4CH 122182156 IC50 > 50000 nM T19244 CQA8B2 122187067 IC50 = 64000 nM T19244 CS5CF1 122187069 IC50 = 12000 nM T19244 C14FGL 122187534 IC50 > 20000 nM T19244 CB7IJ0 122188138 IC50 > 20000 nM T19244 C9TF8M 122190433 IC50 = 25600 nM T19244 C8GHY3 122190972 IC50 > 30000 nM T19244 CTI2V5 122192293 IC50 > 40000 nM T19244 C4NUY0 122192382 IC50 > 10000 nM T19244 C1MVP5 122192989 IC50 = 9089 nM T19244 CLHV68 122192990 IC50 = 22380 nM T19244 C1N0HP 122193176 IC50 > 30000 nM T19244 CV8J6N 122193177 IC50 = 6450 nM T19244 CB8MH7 122193179 IC50 > 30000 nM T19244 CQX7P1 122195090 IC50 > 2000 nM T19244 CUE4R9 122195192 IC50 > 20000 nM T19244 CNF81V 122195193 IC50 > 20000 nM T19244 CCP5U2 122195692 IC50 > 30000 nM T19244 CCP15H 122197303 IC50 = 21000 nM T19244 C1C9LI 122246967 IC50 = 30000 nM T19244 CGT12J 122419159 IC50 > 30000 nM T19244 C2F6EH 122456006 IC50 > 30000 nM T19244 C6QHB4 122484585 IC50 > 50000 nM T19244 COX7E3 122510453 IC50 > 20000 nM T19244 CLM7K3 122604539 IC50 = 29100 nM T19244 C01JHI 122604566 IC50 = 3700 nM T19244 CU2K4P 122650372 IC50 > 10000 nM T19244 C3RCU4 122650378 IC50 = 940 nM T19244 CS47AD 122650581 IC50 = 7400 nM T19244 C5KTB8 122655975 IC50 = 500 nM T19244 CPH1N4 122656020 IC50 = 500 nM T19244 C0VU3O 122656119 IC50 = 1900 nM T19244 C85JKN 122668190 IC50 > 25000 nM T19244 CD6X5P 122669265 IC50 = 10000 nM T19244 C86VYP 122670110 IC50 > 30000 nM T19244 CXP73N 122678088 IC50 = 10000 nM T19244 C1YK2E 122678192 IC50 > 20000 nM T19244 C4P9NG 122700657 EC50 = 34000 nM T19244 CSLF20 123226629 IC50 > 30000 nM T19244 C7ZJ8U 123295297 IC50 > 30000 nM T19244 CT9K0V 124000588 IC50 > 10000 nM T19244 C6CA4O 124088406 IC50 = 2700 nM T19244 C5ZY7L 124114343 IC50 > 50000 nM T19244 CPO7N5 124125214 IC50 = 4600 nM T19244 C4VT3O 124127413 IC50 = 8000 nM T19244 CZEC76 124147932 IC50 > 50000 nM T19244 CEK31I 124148318 IC50 = 2500 nM T19244 C5H2QB 124150512 IC50 > 50000 nM T19244 C6FSR3 124175917 IC50 = 2700 nM T19244 C7TOU4 124175991 IC50 > 10000 nM T19244 CC1O5L 124176023 IC50 = 5900 nM T19244 C49NHK 124176024 IC50 = 2600 nM T19244 C49ONG 124176026 IC50 = 3200 nM T19244 CTD7Q0 124176027 IC50 = 3400 nM T19244 C53AYP 124176028 IC50 > 10000 nM T19244 CB52KW 124176043 IC50 = 1200 nM T19244 CM56CN 124176084 IC50 = 2900 nM T19244 C9RLT1 124176103 IC50 = 7100 nM T19244 CT6HB4 124176198 IC50 = 8700 nM T19244 CL7K0C 124176200 IC50 > 10000 nM T19244 CWMF80 124176201 IC50 = 1800 nM T19244 CYD04K 124176232 IC50 > 10000 nM T19244 CMS9P1 124176233 IC50 > 10000 nM T19244 C7EQH8 124176242 IC50 > 10000 nM T19244 CGJH79 124176281 IC50 > 10000 nM T19244 CCYK63 124176287 IC50 > 10000 nM T19244 CWF7N2 124176288 IC50 > 10000 nM T19244 CK0B3W 124176291 IC50 > 10000 nM T19244 CNC17W 124176295 IC50 > 10000 nM T19244 CMG02Z 124176321 IC50 > 10000 nM T19244 CA3S8B 124221798 IC50 = 850 nM T19244 C3I0PD 124221800 IC50 = 18000 nM T19244 CVKO13 124221803 IC50 = 880 nM T19244 CVI8X5 124221907 IC50 = 510 nM T19244 C84FIJ 124221975 IC50 = 1700 nM T19244 C01UFA 124221976 IC50 = 2300 nM T19244 CDS92J 126483508 IC50 > 50000 nM T19244 CP8W0X 126533801 IC50 > 1000 nM T19244 CIV7R0 126533969 IC50 > 17000 nM T19244 CI97TU 126533981 IC50 > 2000 nM T19244 CIAD86 126534204 IC50 > 20000 nM T19244 C4R7XU 126534291 IC50 > 3000 nM T19244 CVBX50 126534373 IC50 > 3000 nM T19244 CFA3D6 126534516 IC50 > 5000 nM T19244 C0WUJ5 126534771 IC50 > 1000 nM T19244 CX9LM7 126534859 IC50 > 15000 nM T19244 C6DLR7 126534986 IC50 > 1000 nM T19244 C9Q0VB 126535075 IC50 > 16000 nM T19244 CIZC84 126535109 IC50 > 25000 nM T19244 CTAG09 126567264 IC50 > 25000 nM T19244 C5QT4N 126567306 IC50 > 25000 nM T19244 C2LAM7 126591927 IC50 > 30000 nM T19244 CZ3TD0 126651203 IC50 > 50000 nM T19244 C0LTB9 126651349 IC50 > 50000 nM T19244 CS1B2E 127020968 IC50 > 10000 nM T19244 CB2ZK5 127026165 IC50 > 30000 nM T19244 C7J5VX 127026166 IC50 > 30000 nM T19244 C9XU8I 127026167 IC50 > 30000 nM T19244 CU32KG 127026289 IC50 = 1720 nM T19244 CA42BO 127027101 IC50 > 30000 nM T19244 C09CHL 127027102 IC50 > 30000 nM T19244 CCK36V 127029882 IC50 = 3259 nM T19244 CVC84H 127029883 IC50 = 2828 nM T19244 CFY1P0 127029884 IC50 = 397 nM T19244 CU8Y7N 127030224 IC50 = 649 nM T19244 CTEA14 127030225 IC50 = 1562 nM T19244 CLDC46 127031152 IC50 = 16986 nM T19244 C60SMC 127031153 IC50 = 12572 nM T19244 C2POU1 127033963 IC50 > 30000 nM T19244 C2JOP5 127034286 IC50 > 30000 nM T19244 CZ61LK 127034966 IC50 > 10000 nM T19244 CA0SN5 127034967 IC50 > 10000 nM T19244 CWDI07 127037076 IC50 > 20000 nM T19244 C8QIK9 127037551 IC50 > 50000 nM T19244 CI6HK4 127038465 IC50 = 12400 nM T19244 C9Y8VL 127038466 IC50 = 22100 nM T19244 CUBG78 127039139 IC50 > 50000 nM T19244 C60HOC 127040550 IC50 = 40000 nM T19244 C34BGK 127040715 IC50 > 30000 nM T19244 C0J8HC 127041348 IC50 > 3000 nM T19244 CCU4Z1 127041764 IC50 = 26600 nM T19244 CCJX69 127041842 IC50 > 20000 nM T19244 CS78AZ 127041951 IC50 > 30000 nM T19244 CU9C4S 127041952 IC50 > 6000 nM T19244 COW37I 127043420 IC50 = 2100 nM T19244 CVRS53 127043426 IC50 = 13000 nM T19244 C24LTO 127043427 IC50 = 14000 nM T19244 CP42FD 127043428 IC50 = 150 nM T19244 CP25DC 127043607 IC50 = 1400 nM T19244 CQCO27 127046038 IC50 = 2100 nM T19244 C34REM 127046317 IC50 > 30000 nM T19244 C9A1TG 127046557 IC50 = 7200 nM T19244 C57ZRE 127046727 IC50 > 50000 nM T19244 C7YML2 127047647 IC50 > 30000 nM T19244 C48NCK 127047993 IC50 = 2900 nM T19244 C84TQV 127048530 IC50 > 20000 nM T19244 CZV7Q0 127049047 IC50 > 10000 nM T19244 CB54VQ 127049048 IC50 > 10000 nM T19244 C9TUQ2 127049049 IC50 > 10000 nM T19244 CJ8SG3 127049204 IC50 > 50000 nM T19244 CI3X9L 127049803 IC50 = 10990 nM T19244 C2O5LX 127049804 IC50 = 4190 nM T19244 CUVQ34 127050762 IC50 > 50000 nM T19244 CJP90K 127051009 IC50 = 18400 nM T19244 C9V4EG 127051045 IC50 > 50000 nM T19244 C2QX0V 127051283 IC50 = 19000 nM T19244 C7KZJ2 127052145 IC50 > 20000 nM T19244 C38VGB 127052215 IC50 = 13600 nM T19244 CR7O3H 127052463 IC50 = 11800 nM T19244 C4CRE7 127052464 IC50 > 20000 nM T19244 C75EAL 127052638 IC50 > 50000 nM T19244 C2GY5W 127052655 IC50 > 25000 nM T19244 C5OE2H 127053611 IC50 > 20000 nM T19244 CN3XU0 127255875 IC50 > 30000 nM T19244 CEC17N 129164665 IC50 = 11000 nM T19244 CY4B7Z 129164668 IC50 > 50000 nM T19244 CAT90Y 129164701 IC50 = 7000 nM T19244 CUB58Q 129164743 IC50 = 9000 nM T19244 C81SHO 129178830 IC50 = 5000 nM T19244 CJGR20 129240126 IC50 > 30000 nM T19244 CR8HP6 129281194 IC50 > 10000 nM T19244 C7MRB5 129304758 IC50 > 10000 nM T19244 CE8TV5 129893260 IC50 > 25000 nM T19244 C9NPD3 129909153 IC50 > 25000 nM T19244 C4LR9M 129909326 IC50 > 25000 nM T19244 CD80OM 129909338 IC50 = 13200 nM T19244 CV3UP6 129909861 IC50 > 30000 nM T19244 C7WPT8 130301786 IC50 = 150 nM T19244 CK68CA 130453737 IC50 > 30000 nM T19244 CDV84X 131747741 IC50 > 50000 nM T19244 CV06MU 131801402 IC50 = 11900 nM T19244 C4Z5MQ 131839619 IC50 > 30000 nM T19244 CFC05Q 131954513 IC50 = 24700 nM T19244 CN4RF6 132019596 IC50 = 6600 nM T19244 CZ5H2B 132020452 IC50 = 9900 nM T19244 CP8A1Q 132020575 IC50 = 27000 nM T19244 CH8DP7 132220479 IC50 > 20000 nM T19244 C5P4XN 132227197 IC50 > 18000 nM T19244 C1R5SZ 132227201 IC50 > 18000 nM T19244 CGDN94 132275066 IC50 > 10000 nM T19244 CACJ46 132489333 IC50 > 25000 nM T19244 C6Z8BD 132510851 IC50 = 3500 nM T19244 CN12VW 132550264 IC50 = 2360 nM T19244 C9QYP1 132585220 IC50 = 8400 nM T19244 CZC7S8 133081963 IC50 < 5000 nM T19244 C18GQC 134128280 IC50 > 20000 nM T19244 C6DP2E 134130638 IC50 = 200 nM T19244 CS0N2O 134131947 IC50 = 400 nM T19244 CUIF45 134132017 IC50 = 360 nM T19244 CO1RW6 134132142 IC50 > 50000 nM T19244 CB51NS 134133237 IC50 = 1000 nM T19244 CJOQ95 134134229 IC50 = 38300 nM T19244 CES87G 134135247 IC50 = 1445 nM T19244 CDRC75 134136284 IC50 = 3220 nM T19244 CK9MG1 134136380 IC50 = 1800 nM T19244 C5IXF3 134136542 IC50 = 3400 nM T19244 CJ7YU6 134137115 IC50 = 900 nM T19244 CC57VG 134138726 IC50 > 10000 nM T19244 C2A7CZ 134138904 IC50 = 1867 nM T19244 C21OUY 134139520 IC50 > 10000 nM T19244 CU8BV5 134139688 IC50 > 20000 nM T19244 CH3V9Q 134139925 IC50 = 6000 nM T19244 C8MAB7 134142736 IC50 = 5625 nM T19244 CVC1Y4 134142943 IC50 = 6616 nM T19244 C9DBR7 134144418 IC50 > 10000 nM T19244 CK13YN 134145788 IC50 = 8297 nM T19244 C14IWG 134146417 IC50 > 10000 nM T19244 C7DX5U 134148567 IC50 = 450 nM T19244 CFG60Q 134148895 IC50 > 10000 nM T19244 CC43OQ 134149366 IC50 > 50000 nM T19244 CA5B2J 134150245 IC50 = 32970 nM T19244 C0S2VH 134150637 IC50 > 17000 nM T19244 C6NYU2 134150754 IC50 > 5000 nM T19244 C9NI7K 134151534 IC50 = 493 nM T19244 CMTV01 134151719 IC50 > 10000 nM T19244 CZH50T 134151855 IC50 = 3815 nM T19244 C8PT9W 134152052 IC50 > 30000 nM T19244 CP41RT 134154065 IC50 = 20100 nM T19244 CFX51B 134154660 IC50 > 10000 nM T19244 C0LGI2 134154676 IC50 = 2110 nM T19244 CZV9B3 134154775 IC50 = 5210 nM T19244 CQT9F3 134155188 IC50 > 10000 nM T19244 CJ0UG1 134155310 IC50 = 5752 nM T19244 CXT0A2 134155658 IC50 = 340 nM T19244 C9UWD3 134155777 IC50 > 10000 nM T19244 CA49BH 134156727 IC50 > 50000 nM T19244 C7H8GQ 134157229 IC50 > 10000 nM T19244 CNS38M 134157776 IC50 = 5043 nM T19244 CK7B0U 134304087 IC50 > 10000 nM T19244 CX62UZ 134304119 IC50 > 10000 nM T19244 CUDY24 134304129 IC50 > 10000 nM T19244 CO5I4B 134304177 IC50 > 10000 nM T19244 CRD52S 134324842 IC50 > 10000 nM T19244 C17NBC 134325016 IC50 > 10000 nM T19244 CFR87X 134477051 IC50 > 20000 nM T19244 C8W9YN 134477076 IC50 > 20000 nM T19244 CX5MS3 134477080 IC50 > 20000 nM T19244 CSO3Q9 134477081 IC50 > 20000 nM T19244 C51SKX 134477137 IC50 > 20000 nM T19244 CCVX65 134477139 IC50 > 20000 nM T19244 CNU8M6 134477183 IC50 > 20000 nM T19244 CK9SR3 134477213 IC50 > 20000 nM T19244 C1AB5Q 134477222 IC50 > 20000 nM T19244 C9O5FS 134477264 IC50 > 20000 nM T19244 CS5ME8 134477268 IC50 > 20000 nM T19244 CC0OF9 134477275 IC50 > 20000 nM T19244 CVR60G 134539903 IC50 > 25000 nM T19244 C20HAT 134585236 IC50 = 23000 nM T19244 CHA58W 134585452 IC50 = 3000 nM T19244 C6W3VL 134585536 IC50 = 14000 nM T19244 C6Q4RO 134585678 IC50 = 4400 nM T19244 CRL3O8 134585831 IC50 = 29000 nM T19244 CZB7I6 134821685 IC50 > 10000 nM T19244 CDC38O 134823958 IC50 = 2040 nM T19244 CQI48P 135192983 IC50 > 30000 nM T19244 CT0GQ6 135197577 IC50 > 10000 nM T19244 C87VKA 135197594 IC50 > 10000 nM T19244 CQXS07 135197635 IC50 > 10000 nM T19244 C7KXF1 135197643 IC50 > 10000 nM T19244 CS4BM3 135236903 IC50 > 50000 nM T19244 CNEY95 135285657 IC50 = 4000 nM T19244 C2RZN8 135305974 IC50 = 7943.28 nM T19244 CA2OV3 135306913 IC50 > 50000 nM T19244 C8Q4JP 135314141 IC50 < 5000 nM T19244 CW3DO8 135315463 IC50 > 50000 nM T19244 C75MTX 135315494 IC50 > 50000 nM T19244 C7K4PA 135412054 IC50 = 19000 nM T19244 C31VAN 135412231 IC50 = 8800 nM T19244 C9U6OV 135414531 IC50 = 330 nM T19244 C7D6WK 135416383 IC50 = 47000 nM T19244 CX1UD2 135416384 IC50 = 11000 nM T19244 C47LAF 135418940 IC50 > 50000 nM T19244 CIS9K5 135421564 IC50 > 50000 nM T19244 C63ONQ 135435181 IC50 = 840 nM T19244 CZ4GP6 135446244 IC50 > 20000 nM T19244 CFRS56 135446991 IC50 = 5400 nM T19244 CRY8Q1 135453098 IC50 = 2800 nM T19244 CB1M4T 135466520 IC50 = 2200 nM T19244 CWGT82 135502978 IC50 = 26000 nM T19244 CB7S3Y 135530014 IC50 = 345 nM T19244 C3RX6B 135530418 IC50 < 30 nM T19244 CKF13W 135546072 IC50 > 10000 nM T19244 C8R4FB 135546884 IC50 > 20000 nM T19244 CTB8U4 135553266 IC50 = 2900 nM T19244 CL9Q1F 135553267 IC50 = 6600 nM T19244 C6W3AL 135553268 IC50 = 3500 nM T19244 C53HFP 135553269 IC50 = 8100 nM T19244 C5Y6IB 135553271 IC50 = 2800 nM T19244 CY4MV6 135566354 IC50 > 50000 nM T19244 C8DX9H 135567148 IC50 > 25000 nM T19244 C23IWG 135567151 IC50 > 25000 nM T19244 CN1T7U 135681590 IC50 = 91000 nM T19244 CJ4C1Y 135681596 IC50 = 1500 nM T19244 CJZ39U 135681612 IC50 < 40 nM T19244 C3EKM9 135681730 IC50 = 76000 nM T19244 C9UGN1 135681832 IC50 = 100000 nM T19244 C62NOS 135681833 IC50 = 67000 nM T19244 C3D0CJ 135681834 IC50 = 7800 nM T19244 CIG3R9 135681875 IC50 = 47000 nM T19244 CCNH91 135743577 IC50 = 8040 nM T19244 C01PRA 135800176 IC50 = 5700 nM T19244 C62NHL 135800194 IC50 = 42000 nM T19244 C4DH9C 135874529 IC50 = 5100 nM T19244 CSKV72 135883248 IC50 = 6800 nM T19244 CCK5I3 135883253 IC50 = 10000 nM T19244 CC6N5D 135883255 IC50 = 10000 nM T19244 CL5BN6 135883277 IC50 = 10000 nM T19244 C8VL9H 135883279 IC50 = 10000 nM T19244 CDE8Z6 135883307 IC50 = 1700 nM T19244 C94MFR 135883323 IC50 = 2200 nM T19244 CRG82L 135883324 IC50 = 1900 nM T19244 CJ41MZ 135922722 IC50 = 17000 nM T19244 CUX64Z 135922723 IC50 = 8500 nM T19244 C14OBQ 135928469 IC50 > 20000 nM T19244 C01HMT 135932346 IC50 = 20 nM T19244 CT39WL 135938482 IC50 = 6000 nM T19244 C4RL7Q 135985508 IC50 = 800 nM T19244 C1ZT4N 135988927 IC50 = 900 nM T19244 C86BZJ 135988997 IC50 = 1300 nM T19244 C9F1IS 136006171 IC50 = 6400 nM T19244 CEGJ60 136007966 IC50 = 11000 nM T19244 C4HJ7D 136044076 IC50 > 50000 nM T19244 C1SY0D 136045803 IC50 = 1200 nM T19244 CT57ZH 136069450 IC50 > 50000 nM T19244 CFT9R3 136069453 IC50 > 50000 nM T19244 CRPQ42 136069494 IC50 = 65000 nM T19244 CK8Z3V 136069521 IC50 > 50000 nM T19244 CPY1B2 136069522 IC50 > 50000 nM T19244 CX0OM4 136069523 IC50 > 50000 nM T19244 C6EU4D 136069524 IC50 > 50000 nM T19244 CQA2Z1 136069531 IC50 > 50000 nM T19244 CCH31A 136069532 IC50 > 50000 nM T19244 CQ1FS4 136069563 IC50 > 50000 nM T19244 C69JHW 136117992 IC50 < 40 nM T19244 C63VTD 136118015 IC50 = 720 nM T19244 CL08HS 136118016 IC50 = 4000 nM T19244 CTSB03 136118017 IC50 = 2300 nM T19244 CWTZ98 136164050 IC50 = 1700 nM T19244 CGX6C4 136173253 IC50 = 19000 nM T19244 CC52HL 136189674 IC50 > 20000 nM T19244 CQTB32 136205798 IC50 > 10000 nM T19244 CV8QP3 136205832 IC50 > 50000 nM T19244 CB93EM 136205833 IC50 > 50000 nM T19244 CDEX74 136229147 IC50 = 400 nM T19244 CBS97C 136239447 IC50 = 16000 nM T19244 CC8Q2D 136375233 IC50 = 500 nM T19244 C4OVP2 136416802 IC50 > 50000 nM T19244 C7ZCT8 136416815 IC50 > 50000 nM T19244 C95TJH 136632047 IC50 > 50000 nM T19244 CI94YQ 136982007 IC50 > 50000 nM T19244 CK4CM2 137028369 IC50 = 42760 nM T19244 CO6WA9 137313834 IC50 = 560 nM T19244 CE1G4P 137333984 IC50 = 5900 nM T19244 C0PL4B 137434175 IC50 > 30000 nM T19244 C8V9ER 137440575 IC50 = 5300 nM T19244 CS34IR 137628304 IC50 > 25000 nM T19244 C9ACX4 137628305 IC50 > 25000 nM T19244 CP2C1J 137628306 IC50 > 25000 nM T19244 CDGB50 137628309 IC50 > 25000 nM T19244 CW8ZR6 137628310 IC50 < 10000 nM T19244 C48QKY 137628311 IC50 < 10000 nM T19244 CH5AV6 137628312 IC50 > 25000 nM T19244 CU9O3A 137628639 IC50 > 20000 nM T19244 CEZT29 137628641 IC50 > 10000 nM T19244 C6B5US 137628648 IC50 > 10000 nM T19244 C3A6PQ 137628670 IC50 > 10000 nM T19244 C6JO4G 137631841 IC50 > 20000 nM T19244 CES7L0 137632608 IC50 > 20000 nM T19244 CV8M3P 137633531 IC50 < 5000 nM T19244 C28PMQ 137634084 IC50 > 20000 nM T19244 CE9O8V 137634616 IC50 = 1700 nM T19244 CP07AG 137635043 IC50 = 3800 nM T19244 C7S8YV 137636062 IC50 > 20000 nM T19244 CM51CG 137636524 IC50 > 20000 nM T19244 CNA56O 137636856 IC50 > 20000 nM T19244 CH3M0S 137637752 IC50 > 20000 nM T19244 CEN8M3 137638107 IC50 = 4000 nM T19244 CFK9D8 137638117 IC50 > 20000 nM T19244 C8EZ4N 137638256 IC50 > 20000 nM T19244 CLEF51 137638686 IC50 > 20000 nM T19244 C2Y9HF 137638913 IC50 > 20000 nM T19244 C0ZS9N 137638993 IC50 > 20000 nM T19244 CF5TI6 137639661 IC50 = 42100 nM T19244 C5KEW7 137639838 IC50 > 20000 nM T19244 C53ENH 137640507 IC50 > 20000 nM T19244 CN1RV9 137640762 IC50 > 20000 nM T19244 CU0BS2 137641410 IC50 > 20000 nM T19244 CR9C5G 137642830 IC50 <= 20000 nM T19244 CO8V4W 137642907 IC50 > 20000 nM T19244 CJT81N 137643054 IC50 > 20000 nM T19244 CPW7T0 137643121 IC50 = 600 nM T19244 C58ISN 137643139 IC50 = 10000 nM T19244 C1FU3P 137643308 IC50 > 20000 nM T19244 CU91LQ 137644813 IC50 < 5000 nM T19244 C2FOK7 137644816 IC50 > 20000 nM T19244 CN97GA 137645181 IC50 > 50000 nM T19244 C5UL6D 137645197 IC50 > 20000 nM T19244 CNB72K 137645644 IC50 > 20000 nM T19244 C9Q0MH 137645867 IC50 = 580 nM T19244 CH0TP2 137645931 IC50 > 20000 nM T19244 CU47YW 137646415 IC50 > 20000 nM T19244 C5IHS8 137646440 IC50 > 20000 nM T19244 CN4U1A 137646732 IC50 > 30000 nM T19244 CDCH19 137646766 IC50 > 20000 nM T19244 CLT73G 137647199 IC50 > 10000 nM T19244 CE57QM 137647529 IC50 > 20000 nM T19244 CGW71J 137647660 IC50 > 50000 nM T19244 CP32AR 137648836 IC50 > 20000 nM T19244 C5AT7D 137649062 IC50 > 20000 nM T19244 CYU2J5 137649494 IC50 > 20000 nM T19244 C04JSE 137649716 IC50 = 7500 nM T19244 C8N9CH 137650363 IC50 = 710 nM T19244 C2JBS1 137651899 IC50 > 100000 nM T19244 CV4AP0 137652684 IC50 > 20000 nM T19244 CKV03G 137653074 IC50 > 30000 nM T19244 C38FXZ 137653443 IC50 > 20000 nM T19244 CV59RY 137654290 IC50 < 5000 nM T19244 CSRK73 137655508 IC50 = 60000 nM T19244 C17LIA 137655641 IC50 > 33000 nM T19244 CJ7D8K 137655914 IC50 > 20000 nM T19244 C1OXG8 137655944 IC50 > 10000 nM T19244 CTW5P4 137656265 IC50 > 20000 nM T19244 CZ4W3T 137656391 IC50 > 50000 nM T19244 CU28CY 137657424 IC50 > 20000 nM T19244 CB61UY 137658460 IC50 > 20000 nM T19244 CG96FH 137658637 IC50 > 50000 nM T19244 C9VOB4 137658779 IC50 > 20000 nM T19244 CJ8L1W 137659170 IC50 = 33 nM T19244 CH4M3X 137659806 IC50 > 20000 nM T19244 CF8HN9 137661762 IC50 > 20000 nM T19244 C0XCS4 137661956 IC50 > 20000 nM T19244 C96QPV 137662004 IC50 = 2500 nM T19244 CFC3L4 137662114 IC50 > 20000 nM T19244 C6KYD7 137700754 IC50 > 10000 nM T19244 CJC95O 138319684 IC50 = 25000 nM T19244 CPTE92 138319693 IC50 = 135 nM T19244 CE79SV 138377584 IC50 > 50000 nM T19244 CB8FE3 138393376 IC50 > 5000 nM T19244 CKDZ26 138504497 IC50 > 30000 nM T19244 C1XSH7 138594194 IC50 > 10000 nM T19244 CG4RO6 138632227 IC50 > 18000 nM T19244 CHT39X 138632268 IC50 > 18000 nM T19244 CVB6L2 138632650 IC50 > 18000 nM T19244 CI9YB7 138753112 IC50 = 21400 nM T19244 CJA5H2 138756812 IC50 >= 20000 nM T19244 C1BOT2 139030270 IC50 = 2700 nM T19244 CD29IP 139507088 IC50 > 10000 nM T19244 CF8LN1 139582020 IC50 > 30000 nM T19244 CI1D9F 139600335 IC50 = 78100 nM T19244 CG2NH6 139600336 IC50 = 9900 nM T19244 C0HN5J 139600337 IC50 = 4400 nM T19244 C2K4QW 140251527 IC50 < 10000 nM T19244 CU2ND3 140251533 IC50 < 10000 nM T19244 CGA12N 141473855 IC50 = 3380 nM T19244 C2YC6F 141473885 IC50 = 3930 nM T19244 C9JSZ2 141529337 IC50 > 10000 nM T19244 CSE1D2 141529338 IC50 > 10000 nM T19244 C43LDR 141730928 IC50 > 50000 nM T19244 C17XZS 142727681 IC50 = 3500 nM T19244 C1UCX0 144953608 IC50 > 10000 nM T19244 C9GRB2 144953612 IC50 > 10000 nM T19244 CV4X5P 144953614 IC50 > 10000 nM T19244 C1W8QR 145865307 IC50 = 1990 nM T19244 C9ISH6 145925685 IC50 = 17000 nM T19244 CF1MH2 145949267 IC50 > 30000 nM T19244 CXJ07F 145949470 IC50 > 50000 nM T19244 CI3V6Y 145950358 IC50 = 36000 nM T19244 CLZ54T 145950740 IC50 = 32000 nM T19244 C4FM3C 145951105 IC50 > 50000 nM T19244 CLV0G6 145951167 IC50 = 36000 nM T19244 CH0K8V 145951521 IC50 = 2200 nM T19244 CG5OW3 145951998 IC50 = 48000 nM T19244 CEB71V 145952023 IC50 > 30000 nM T19244 C4LJV9 145952024 IC50 = 43000 nM T19244 C1QA6W 145952070 IC50 = 59000 nM T19244 CC7IP8 145952109 IC50 = 6300 nM T19244 CN0S3B 145952357 IC50 = 1600 nM T19244 C3E5BK 145952508 IC50 > 10000 nM T19244 C0RGQ7 145952699 IC50 > 10000 nM T19244 C9D5MZ 145952745 IC50 = 28000 nM T19244 CRN85T 145952991 IC50 > 25000 nM T19244 CA7W2O 145953059 IC50 = 19000 nM T19244 C5LB7M 145953999 IC50 = 28000 nM T19244 CW9I0R 145954143 IC50 > 10000 nM T19244 CN5L4K 145954640 IC50 = 4800 nM T19244 CWA8H2 145955288 IC50 > 30000 nM T19244 CQ5SN1 145955289 IC50 = 4400 nM T19244 C7N6CA 145956935 IC50 = 6100 nM T19244 CBFU43 145957229 IC50 = 16000 nM T19244 C20EDK 145957568 IC50 = 23000 nM T19244 CFZJ34 145957574 IC50 > 19952.62 nM T19244 C3B0YE 145957778 IC50 = 2800 nM T19244 CID3G5 145958087 IC50 > 50000 nM T19244 CM8U9A 145958674 IC50 = 2000 nM T19244 CBF54O 145958967 IC50 > 50000 nM T19244 CB5XW7 145959080 IC50 = 2600 nM T19244 CLS3W5 145959177 IC50 > 25000 nM T19244 CLJE41 145959897 IC50 > 25000 nM T19244 CW1GO5 145960043 IC50 = 3000 nM T19244 CDKY72 145960338 IC50 > 50000 nM T19244 CT6OH1 145960389 IC50 > 50000 nM T19244 CZ83QK 145960490 IC50 > 50000 nM T19244 C0WB6J 145960881 IC50 > 20000 nM T19244 C5ZD1H 145961500 IC50 > 30000 nM T19244 C42PLT 145962320 IC50 > 100000 nM T19244 CDY47R 145962388 IC50 > 50000 nM T19244 CQ2TN4 145962919 IC50 = 27000 nM T19244 CKLA91 145962920 IC50 = 8500 nM T19244 C62MVS 145964029 IC50 = 500 nM T19244 CFAK41 145964101 IC50 = 25000 nM T19244 C2IM3V 145964416 IC50 = 5000 nM T19244 CRZ5T1 145964880 IC50 > 10000 nM T19244 C7SK5V 145965195 IC50 > 10000 nM T19244 CSK8Y1 145965486 IC50 = 11800 nM T19244 C4P7UD 145965756 IC50 = 200 nM T19244 C2MS3R 145966170 IC50 >= 30000 nM T19244 CRS65V 145966585 IC50 > 10000 nM T19244 CW02FZ 145967133 IC50 = 8000 nM T19244 CC0QA2 145967606 IC50 = 13000 nM T19244 C19IVD 145967885 IC50 = 14000 nM T19244 CX42BV 145968371 IC50 > 50000 nM T19244 CG2A0S 145968399 IC50 > 50000 nM T19244 CU6RH3 145968879 IC50 > 50000 nM T19244 CJUK65 145968931 IC50 > 10000 nM T19244 CCB21N 145969176 IC50 > 10000 nM T19244 CA12HV 145969294 IC50 = 19000 nM T19244 C4HF5M 145969366 IC50 = 100 nM T19244 C94URS 145969597 IC50 = 100 nM T19244 C2S8DE 145969909 IC50 = 4400 nM T19244 CI3O2K 145970611 IC50 > 20000 nM T19244 C6CD4Z 145970793 IC50 = 17000 nM T19244 CS5U3M 145970807 IC50 = 15000 nM T19244 C1RCP7 145972319 IC50 < 10000 nM T19244 CXF9E7 145972420 IC50 = 2900 nM T19244 CV9OM2 145973260 IC50 > 10000 nM T19244 C8RFM3 145973261 IC50 > 20000 nM T19244 C6OI3K 145973962 IC50 > 10000 nM T19244 C4XZ1W 145973987 IC50 = 200 nM T19244 C56HYE 145974067 IC50 = 28000 nM T19244 CJN96Q 145974556 IC50 > 50000 nM T19244 CGWM29 145974840 IC50 = 16500 nM T19244 CAU82Y 145975252 IC50 > 10000 nM T19244 CSBQ67 145975261 IC50 > 10000 nM T19244 CUZ47S 145975654 IC50 > 10000 nM T19244 CQ2H6F 145976125 IC50 > 10000 nM T19244 CUV49K 145977796 IC50 = 5700 nM T19244 C4XV7J 145978553 IC50 > 10000 nM T19244 C3S0UI 145978581 IC50 = 11900 nM T19244 CWA6L3 145981037 IC50 > 20000 nM T19244 CGA83C 145981271 IC50 > 10000 nM T19244 CJ35DM 145984299 IC50 = 100000 nM T19244 C4HAP0 145984727 IC50 > 25000 nM T19244 C5R6BS 145987142 IC50 > 10000 nM T19244 C7O1PF 145987480 IC50 = 14000 nM T19244 C81LEH 145987485 IC50 > 20000 nM T19244 CMRQ02 145987862 IC50 > 20000 nM T19244 C7GK3H 145990715 IC50 = 60500 nM T19244 CE1L5T 145992719 IC50 > 20000 nM T19244 CMIH10 145993513 IC50 > 20000 nM T19244 C8X2IT 145996536 IC50 > 50000 nM T19244 CHJ79V 145997874 IC50 > 10000 nM T19244 CAU3Z1 146020618 IC50 = 4000 nM T19244 CZE16B 146026197 IC50 > 50000 nM T19244 C7F6SU 146047134 IC50 > 200000 nM T19244 CBRE71 146047136 IC50 > 20000 nM T19244 C2RJ1U 146176418 IC50 = 46600 nM T19244 CS54CM 146433251 IC50 > 40000 nM T19244 CGO5C4 146433253 IC50 > 40000 nM T19244 C61LGO 146433463 IC50 > 40000 nM T19244 C4OSN5 146433538 IC50 > 40000 nM T19244 CN2MA4 146433574 IC50 > 40000 nM T19244 C5ZOJ3 146680920 IC50 > 100000 nM T19244 C9YJZ5 147180858 IC50 = 8370 nM T19244 CUAY08 148018738 IC50 > 10000 nM T19244 CQK39B 149491764 IC50 > 10000 nM T19244 C1ZX5D 149494192 IC50 > 10000 nM T19244 CL6T4P 149986651 IC50 > 20000 nM T19244 CTI5R1 151961601 IC50 = 13400 nM T19244 CC3ME1 152131905 IC50 = 18000 nM T19244 C36ISR 153434865 IC50 > 10000 nM T19244 CG5IF7 154701259 IC50 > 1000 nM T19244 C2J9YV 154727580 IC50 = 330000 nM T19244 CZE1S5 155126870 IC50 > 50000 nM T19244 CI6EB5 155126882 IC50 > 50000 nM T19244 CF2CU8 155510758 IC50 > 30000 nM T19244 CG5HO8 155511239 IC50 > 100000 nM T19244 C7ZE5Q 155511547 IC50 = 16000 nM T19244 CQ83KZ 155512662 IC50 > 10000 nM T19244 CT74QE 155513632 IC50 = 1500 nM T19244 CPE58H 155514125 IC50 = 19000 nM T19244 CD53LC 155514863 IC50 > 25000 nM T19244 CMZ4Q7 155515478 IC50 > 25000 nM T19244 CDV4Z6 155515709 IC50 = 1940000 nM T19244 CCJ14L 155516448 IC50 = 300 nM T19244 C49INQ 155516757 IC50 > 50000 nM T19244 CA3K9P 155517032 IC50 < 10000 nM T19244 CRD79Z 155518589 IC50 = 10000 nM T19244 C30SPO 155518654 IC50 > 50000 nM T19244 C28HEF 155519544 IC50 > 100000 nM T19244 C0KLD8 155519559 IC50 > 100000 nM T19244 CI9U3X 155521508 IC50 = 8300 nM T19244 CK7RM1 155521671 IC50 >= 20000 nM T19244 CGQ1X0 155522363 IC50 = 9300 nM T19244 C0ZXV4 155522886 IC50 > 25000 nM T19244 CWCN51 155522922 IC50 > 50000 nM T19244 CC5GO1 155523088 IC50 = 22300 nM T19244 C2LO4Y 155523731 IC50 > 25000 nM T19244 C3LC2H 155523754 IC50 > 20000 nM T19244 C12KNB 155523817 IC50 = 480 nM T19244 CYI71L 155523951 IC50 = 15900 nM T19244 CTU67Z 155524559 IC50 > 100000 nM T19244 CG71WI 155525128 IC50 > 25000 nM T19244 CI31SP 155527821 IC50 = 6000 nM T19244 C05QTC 155528035 IC50 > 25000 nM T19244 C5QA2B 155529241 IC50 < 10000 nM T19244 C9U8FN 155529326 IC50 = 9400 nM T19244 C7SEX2 155529894 IC50 = 5400 nM T19244 C4F7WU 155530183 IC50 = 17020 nM T19244 CQ6F7O 155530369 IC50 > 25000 nM T19244 CFL61W 155532250 IC50 = 12300 nM T19244 C63HSA 155534748 IC50 = 20000 nM T19244 C3F8NR 155536006 IC50 = 7943.28 nM T19244 C8K3XJ 155537606 IC50 > 20000 nM T19244 CM3PB2 155537682 IC50 > 25000 nM T19244 CCO96S 155538113 IC50 = 9000 nM T19244 CDU52V 155538567 IC50 = 260 nM T19244 CUS3I9 155538644 IC50 < 10000 nM T19244 C1FZY9 155539610 IC50 = 4490 nM T19244 CGH8T5 155540333 IC50 = 6600 nM T19244 CB43YR 155540395 IC50 > 40000 nM T19244 C5T9KE 155542416 IC50 > 50000 nM T19244 CNH46F 155543687 IC50 > 40000 nM T19244 C57ICR 155544322 IC50 = 5011.87 nM T19244 C8WGH1 155544876 IC50 = 5011.87 nM T19244 CV13XI 155546721 IC50 = 6309.57 nM T19244 CQ6D2C 155547369 IC50 > 25000 nM T19244 CRY3A2 155548898 IC50 > 30000 nM T19244 CH25ZD 155549064 IC50 > 50000 nM T19244 CJD38X 155549583 IC50 > 25000 nM T19244 CHDG36 155550819 IC50 > 25000 nM T19244 CUH7R2 155553391 IC50 > 10000 nM T19244 C7JCS2 155553955 IC50 > 25000 nM T19244 C7N5HA 155554052 IC50 = 22600 nM T19244 C8Q2FG 155555556 IC50 > 20000 nM T19244 C09FGY 155555863 IC50 > 25000 nM T19244 CIK75H 155556042 IC50 > 25000 nM T19244 C3WT2Q 155556441 IC50 > 50000 nM T19244 C9H1VK 155556442 IC50 > 50000 nM T19244 CQB48L 155556931 IC50 = 17200 nM T19244 CNH27R 155557555 IC50 > 20000 nM T19244 C4HPK2 155558743 IC50 > 25000 nM T19244 CKZT21 155559364 IC50 > 20000 nM T19244 CEF9N6 155560028 IC50 = 10000 nM T19244 CF4LM6 155560880 IC50 < 10000 nM T19244 CM7ZG9 155561160 IC50 > 25000 nM T19244 C9HIU5 155561551 IC50 = 10000 nM T19244 C1MW3L 155561646 IC50 = 17800 nM T19244 CL3A2S 155562076 IC50 = 1900 nM T19244 CKX10W 155562129 IC50 = 20480 nM T19244 C6T2RV 155562253 IC50 < 10000 nM T19244 CCOD50 155562467 IC50 = 14400 nM T19244 CFVB79 155562854 IC50 = 82000 nM T19244 CG95WV 155563831 IC50 > 20000 nM T19244 CWOE21 155564042 IC50 > 30000 nM T19244 CMK03D 155564568 IC50 < 10000 nM T19244 CC5FE7 155564581 IC50 > 50000 nM T19244 CIBA72 155564665 IC50 = 20300 nM T19244 CK9N0Z 155567885 IC50 > 10000 nM T19244 CMC2A9 155568311 IC50 > 50000 nM T19244 CKYJ21 76283430 IC50 > 20000 nM T19244 CIJ3N0 76283682 IC50 > 30000 nM T19244 D00AEX 44341439 IC50 > 100000 nM T19244 D00AWM 9826520 IC50 > 10000000 nM T19244 D00EMF 3644637 IC50 > 100000 nM T19244 D00PYW 44341256 IC50 = 1810 nM T19244 D00XDG 11708263 IC50 > 50000 nM T19244 D00YNA 25093374 IC50 = 2100 nM T19244 D01ARE 44388719 IC50 = 2100 nM T19244 D01JFF 44191096 IC50 > 30000 nM T19244 D01JPJ 66731056 IC50 > 10000 nM T19244 D01UYI 5281607 IC50 = 5225 nM T19244 D01YWE 25207521 IC50 = 6500 nM T19244 D02BGR 9949648 IC50 = 5300 nM T19244 D02DEF 49765871 IC50 = 11000 nM T19244 D02DTR 44341278 IC50 = 185 nM T19244 D02EAP 11993867 Ki = 1300 nM T19244 D02GFK 25034431 IC50 = 48970 nM T19244 D02HNQ 46182736 IC50 = 4000 nM T19244 D02KZD 71598521 IC50 = 7400 nM T19244 D02TSN 46244454 IC50 > 10000 nM T19244 D03KXT 44341260 IC50 = 101 nM T19244 D03NMM 46843035 IC50 = 4500 nM T19244 D03YHZ 25147692 IC50 = 2900 nM T19244 D04VPH 45376872 IC50 > 30000 nM T19244 D05EMX 14076674 Ki = 2000 nM T19244 D05MSG 44593666 IC50 > 40000 nM T19244 D05NWH 443390 IC50 = 82000 nM T19244 D05VQJ 25147749 IC50 > 10000 nM T19244 D05XGR 6918647 IC50 > 100000 nM T19244 D06CWR 24754344 IC50 = 1270 nM T19244 D06EMC 11392888 IC50 > 30000 nM T19244 D06HOI 44249821 IC50 = 29200 nM T19244 D06MBD 11176403 IC50 > 10000 nM T19244 D06QFO 11332763 Ki = 5900 nM T19244 D06TRS 23646069 Ki = 46600 nM T19244 D06UEP 17027464 IC50 > 25000 nM T19244 D06VDN 443391 IC50 = 23000 nM T19244 D07ADX 54764565 IC50 > 30000 nM T19244 D07ANY 1367 IC50 = 42900 nM T19244 D07GCA 11514705 IC50 > 10000 nM T19244 D07VHB 11321889 IC50 = 96 nM T19244 D07WLT 25180108 IC50 = 28300 nM T19244 D08HUX 3530525 IC50 = 30000 nM T19244 D08IDC 24827305 IC50 = 1888 nM T19244 D08QPU 72737723 IC50 = 4800 nM T19244 D08UWZ 16725047 IC50 > 40000 nM T19244 D08ZYC 11595431 IC50 > 33000 nM T19244 D09CPC 13728862 IC50 = 58900 nM T19244 D09PTP 57325421 IC50 > 10000 nM T19244 D09ZPN 135416394 IC50 = 39000 nM T19244 D0A0GU 44247568 IC50 > 10000 nM T19244 D0AS0V 10141 IC50 > 10000 nM T19244 D0B0LC 44341428 IC50 = 130 nM T19244 D0BD6A 10278617 IC50 > 10000 nM T19244 D0BU8W 44219611 IC50 > 100000 nM T19244 D0BV3B 16214871 IC50 > 30000 nM T19244 D0D3CJ 10308091 IC50 = 3162.28 nM T19244 D0DA1E 23642319 IC50 > 10000 nM T19244 D0DY5G 443389 IC50 > 100000 nM T19244 D0F5EI 10017019 IC50 > 10000 nM T19244 D0G3TK 5280863 Ki = 6000 nM T19244 D0G6BJ 24802842 IC50 = 10000 nM T19244 D0G9WP 18407230 IC50 = 123000 nM T19244 D0G9YL 16214849 IC50 = 17000 nM T19244 D0H1OK 11562302 IC50 > 100000 nM T19244 D0I7GE 11790 IC50 > 10000 nM T19244 D0IM5E 11450263 IC50 > 100000 nM T19244 D0J0TP 9917862 IC50 > 30000 nM T19244 D0J1IE 11993873 Ki = 14100 nM T19244 D0J1QT 44473100 IC50 > 40000 nM T19244 D0J4CB 24803184 IC50 = 8000 nM T19244 D0J6RQ 6437306 IC50 = 1800 nM T19244 D0JD4C 9853498 IC50 = 200 nM T19244 D0K3EW 49799108 IC50 = 3000 nM T19244 D0K4LS 10691533 IC50 = 59000 nM T19244 D0L2WP 46225540 IC50 = 500 nM T19244 D0M0IQ 11210706 IC50 = 710 nM T19244 D0M4SY 135440466 IC50 = 1200 nM T19244 D0N2KU 44517677 IC50 > 30000 nM T19244 D0N4LR 53469448 IC50 = 4500 nM T19244 D0NM0P 25093389 IC50 = 800 nM T19244 D0O1HH 11263510 Ki = 1200 nM T19244 D0O8WT 10338547 IC50 = 600 nM T19244 D0P0IE 10205 IC50 > 10000 nM T19244 D0P8PK 10192730 IC50 = 1050 nM T19244 D0PC5A 44243144 IC50 > 10000 nM T19244 D0Q0PN 11494579 IC50 = 18000 nM T19244 D0R0IB 56587994 IC50 > 30000 nM T19244 D0R0TW 11964036 IC50 > 10000 nM T19244 D0R2TW 10238338 IC50 = 14000 nM T19244 D0S0QN 1712706 IC50 = 45603691.6 nM T19244 D0S6GE 5327067 IC50 = 11000 nM T19244 D0S9CI 11989776 IC50 > 30000 nM T19244 D0U7BJ 44341234 IC50 = 129 nM T19244 D0U7OD 16043230 IC50 > 30000 nM T19244 D0V0YM 24871527 IC50 = 18000 nM T19244 D0V2QH 24894072 IC50 = 1640 nM T19244 D0V3ZG 25192022 IC50 = 3900 nM T19244 D0V4EX 54760053 IC50 > 40000 nM T19244 D0VD5O 11148236 Ki > 400000 nM T19244 D0W3XD 16049828 IC50 > 30000 nM T19244 D0WU1S 52912189 IC50 = 9900 nM T19244 D0Y1YR 442793 IC50 = 12100 nM T19244 D0Y4BL 11676971 IC50 > 10000 nM T19244 D0YM4A 22319604 IC50 > 10000 nM T19244 D0YP4A 11993866 Ki = 400 nM T19244 D0YQ8U 11993871 Ki = 900 nM T19244 D0YQ8V 46236221 IC50 > 30000 nM T19244 D0YW6B 44627267 IC50 = 3700 nM T19244 D0ZY7X 697226 IC50 > 5000 nM T36059 D04JEE 4946 EC50 > 5011.87 nM T36059 D04OSE 4485 Ki = 8290 nM T36059 D06IAR 60961 IC50 = 1.148 nM T36059 D09AMZ 1676 Ki = 92600 nM T36059 D0B3HD 2519 Ki > 13300 nM T36059 D0F8RA 2153 Ki = 14 nM T36059 D0K8KX 5280343 Ki = 30000 nM T36059 D0T0KA 4474 Ki = 3250 nM T36059 D0XE1C 219024 Ki > 10 nM T36059 D00OAU 9869857 EC50 = 4.2 nM T36059 D00SUK 216466 Ki > 10000 nM T36059 D02YQO 10668061 Ki > 10000 nM T36059 D03OQI 11618368 Ki = 1570 nM T36059 D07TEP 10117987 Ki > 1000 nM T36059 D09TFB 9896267 IC50 = 4800 nM T36059 D0B4VE 10251 Ki = 50100 nM T36059 D0F4ZY 5311037 Ki > 3000 nM T36059 D0F5UN 9953065 Ki = 200 nM T36059 D0G4CF 11270783 Ki = 1070 nM T36059 D0L5VS 6448585 Ki = 2500 nM T36059 D0L9KH 44623998 IC50 = 3300 nM T36059 D0LI1C 44469321 IC50 = 8300 nM T36059 D0QG9A 9805430 Ki = 45 nM T36059 D0U0KR 3035850 Ki = 0.2 nM T36059 D0X0IY 64627 Ki = 4390 nM T36059 D0Y6ZK 123683 IC50 = 0.02291 nM T36059 D0Z3PO 21874557 Ki = 1005 nM T36059 D0Z9RJ 11561692 Ki > 1000 nM T36059 D08ECB 11716665 Ki > 1000 nM T36059 D0I5VA 11248240 Ki = 0.29 nM T36059 D00YSJ 158795 Ki = 25800 nM T36059 D01VPK 6439091 Ki = 2800 nM T36059 D07ESH 176408 Ki > 1000 nM T36059 D0B1MJ 6918097 Ki = 1900 nM T36059 D0E4WF 439176 Ki = 680 nM T36059 D0J2UW 3086599 EC50 = 10 nM T36059 D0NQ5I 65710 Ki = 47 nM T36059 D0V5DX 9884817 Ki = 2511.89 nM T36059 D0Y6GJ 176407 Ki = 300 nM T36059 C7B8VJ 44405080 Ki = 3.7 nM T36059 CF92BM 45482610 EC50 = 2.8 nM T36059 C3CJS6 1330 Ki = 183 nM T36059 C32LCX 3545 Ki = 25000 nM T36059 CHE7P9 8975 Ki = 99 nM T36059 CX0YR8 20345 Ki = 22 nM T36059 C28VFY 60602 Ki = 2800 nM T36059 CNM9L6 65102 Ki = 75 nM T36059 CKF52M 71593 Ki > 100000 nM T36059 CS4QG5 92208 Ki = 41.3 nM T36059 C3SPQ5 95121 Ki > 100000 nM T36059 C2CG8M 98567 Ki = 6.4 nM T36059 C4VE6D 99562 Ki > 10000 nM T36059 CGB03T 102175 Ki = 9.3 nM T36059 CC90DA 102213 IC50 = 15 nM T36059 C57IVM 126054 Ki = 12.4 nM T36059 C6OGM1 131432 Ki = 54.2 nM T36059 C2J0SC 131450 Ki = 578 nM T36059 CU7A5O 149362 IC50 = 104 nM T36059 C8ZM5K 165506 Ki = 42800 nM T36059 CF59MP 169662 Ki = 297 nM T36059 C0X8NW 176925 Ki = 6070 nM T36059 CL08HI 185566 Ki > 100000 nM T36059 C73MBU 197637 Ki = 41 nM T36059 CA6E5H 215492 Ki = 9450 nM T36059 CD0MT5 215610 Ki = 32 nM T36059 C2L5UM 252744 Ki = 5240 nM T36059 CFO07N 254343 Ki = 50100 nM T36059 CGYS02 282663 Ki = 2510 nM T36059 CMH1F9 308531 Ki = 14000 nM T36059 C5BK1O 314836 Ki > 1000 nM T36059 CSZ1R6 317946 Ki > 9000 nM T36059 CCO63F 354785 Ki = 48000 nM T36059 C4PY5W 355189 Ki = 12000000 nM T36059 CLZE79 386674 Ki > 10000 nM T36059 C0QG9C 447594 Ki = 301 nM T36059 C58QWF 456309 Ki = 6941 nM T36059 CJ64SM 462569 Ki = 1300000 nM T36059 CPL8Z1 463104 Ki = 2300000 nM T36059 C4JE9F 463105 Ki = 730 nM T36059 C3PRE8 463106 Ki = 310000 nM T36059 CE69BJ 463107 Ki = 980000 nM T36059 C96QNP 495847 Ki >= 10000 nM T36059 C9GZ0J 541903 Ki = 816 nM T36059 CI0CW2 570244 Ki = 300 nM T36059 C7PN9X 604454 Ki = 22000 nM T36059 CSV78R 626711 Ki = 8020 nM T36059 C0QI3X 627207 Ki = 1380 nM T36059 CML1Z5 631095 Ki = 3370 nM T36059 C93YWM 634113 Ki = 16200 nM T36059 CB41OV 639625 Ki = 3900000 nM T36059 CAH8B6 639626 Ki = 15000000 nM T36059 CV2D4A 640847 Ki = 950 nM T36059 CXJ93T 640935 Ki = 35000000 nM T36059 CY3H8D 832542 Ki = 9900 nM T36059 CXGJ45 845925 Ki = 27000000 nM T36059 CUXB69 846029 Ki = 2600000 nM T36059 C8Y4NV 851050 Ki > 10000 nM T36059 CC94MT 851051 Ki > 10000 nM T36059 CCM2J1 851052 Ki > 10000 nM T36059 CNJC61 853426 Ki = 440 nM T36059 CHJV30 906099 Ki > 1000 nM T36059 C5QFM2 933735 IC50 > 10000 nM T36059 CFW26I 980118 Ki = 887 nM T36059 CWME72 982689 Ki = 1000 nM T36059 C75YIZ 1006361 Ki = 770 nM T36059 C75VMR 1047282 IC50 = 186 nM T36059 CO2SD9 1076689 IC50 = 5760 nM T36059 CIBE02 1203667 Ki = 5600000 nM T36059 C8ZM4G 1241166 Ki > 1000 nM T36059 C5P2TF 1487654 Ki > 1000 nM T36059 CI5J9A 1487656 Ki > 1000 nM T36059 CM80QJ 1509337 Ki > 10000 nM T36059 CLU5E8 1899510 Ki = 177 nM T36059 CLI97S 2241546 Ki = 140 nM T36059 C0G5JB 2241547 Ki = 520 nM T36059 C3I9YT 2440996 Ki = 2800 nM T36059 C3ZP1T 2539471 Ki = 2100 nM T36059 CJB2C5 2660435 Ki = 1800 nM T36059 C8L6SZ 2660552 Ki = 3700 nM T36059 CK8T0W 2748282 Ki > 10000 nM T36059 CWY03R 2778758 Ki = 35800 nM T36059 CW3Z7Q 2814825 Ki > 1000 nM T36059 C5OKU7 2820730 Ki = 13000 nM T36059 CV5L2P 2847113 Ki = 12000 nM T36059 CL0U6S 2847148 Ki = 5900 nM T36059 CZJ51C 2848828 IC50 = 255 nM T36059 CN9C6E 2861880 IC50 = 407 nM T36059 C51GNW 2874872 Ki > 10000 nM T36059 CHWU72 2910343 Ki = 5060 nM T36059 CS6Q9H 2989397 Ki > 100000 nM T36059 CRO73B 2989630 Ki = 13300 nM T36059 CWMB15 3042985 Ki = 85.3 nM T36059 C5TCF2 3044933 Ki = 44 nM T36059 CBM9N7 3071852 Ki = 489 nM T36059 CC48UQ 3162481 Ki > 10000 nM T36059 C2GE9F 3162506 Ki > 10000 nM T36059 C4ZI9K 3162667 Ki > 1000 nM T36059 CH5L8S 3359650 Ki > 1000 nM T36059 CZD52B 3462248 Ki = 3200 nM T36059 CB7A6X 3462249 Ki = 3500 nM T36059 CYHO51 3534313 Ki = 4600 nM T36059 CR7H8U 4066469 Ki = 11000000 nM T36059 C0O1QY 4247733 Ki = 300 nM T36059 CPW02K 4885273 Ki = 300 nM T36059 CTG1E3 5002053 Ki = 3200 nM T36059 C70ILQ 5033052 Ki = 208 nM T36059 C7FYA5 5078908 Ki = 48000000 nM T36059 CZB37F 5311431 Ki = 915 nM T36059 C49DTY 5364053 Ki = 4140 nM T36059 C4ACV8 5368229 Ki = 72.4 nM T36059 CWUL54 5378171 Ki = 6700 nM T36059 CB6O5S 5458461 Ki = 4590 nM T36059 CB49EP 5836591 Ki = 23000 nM T36059 CGAX04 6436223 Ki = 1080 nM T36059 CTK1P2 6439089 Ki = 30 nM T36059 CMQ01S 6480505 Ki = 40.3 nM T36059 CGB63D 6604881 Ki = 2770 nM T36059 C5L8EP 7214067 Ki > 10000 nM T36059 C2TX5N 7315332 Ki = 487 nM T36059 C0B8TL 8924077 Ki = 2500 nM T36059 C70MOW 9246778 Ki = 1500 nM T36059 C3O8GK 9247074 Ki = 3200 nM T36059 CVK1H5 9247113 Ki = 1000 nM T36059 C7BR3G 9799990 Ki = 466 nM T36059 CKNT38 9801343 Ki = 0.2 nM T36059 C2VPI6 9802080 Ki = 55.1 nM T36059 C0BJD9 9803226 Ki > 6 nM T36059 CRHL94 9803956 Ki = 15 nM T36059 C6J2LD 9803966 Ki = 18.1 nM T36059 C2EJD7 9803992 Ki = 25 nM T36059 C5V4ZC 9804259 Ki = 193 nM T36059 C92LUT 9805713 EC50 = 0.7 nM T36059 C98ERU 9814428 Ki = 760 nM T36059 CZR3N8 9816781 Ki = 425 nM T36059 C0JI5S 9819926 Ki = 2511.89 nM T36059 CVLM89 9821879 Ki = 170 nM T36059 C0VBX9 9822083 Ki = 17500 nM T36059 C0TS3U 9822488 Ki = 1000 nM T36059 C2O9IQ 9822747 Ki = 0.4 nM T36059 CU5V3E 9824370 Ki = 395 nM T36059 CAQS87 9824812 Ki = 0.7998 nM T36059 CK0FX6 9825550 Ki = 137 nM T36059 C3YK7B 9825923 Ki = 50.5 nM T36059 CUG62V 9827467 Ki > 5000 nM T36059 CP04RO 9828174 Ki = 16 nM T36059 CNM9W5 9828356 EC50 = 3.4 nM T36059 C9BZC8 9836304 Ki = 1291 nM T36059 CS6IN9 9839378 Ki = 23 nM T36059 CFXZ58 9839545 Ki = 30.8 nM T36059 CK1FP4 9840375 Ki = 20 nM T36059 C6IH2G 9841022 Ki = 2270 nM T36059 C4TOH3 9841364 Ki = 1100 nM T36059 CZ7Y9F 9841369 Ki = 1870 nM T36059 C25KVI 9842054 Ki = 540 nM T36059 C7L8SQ 9842502 Ki = 15300 nM T36059 C12UDF 9843101 Ki = 0.4 nM T36059 CGB16Y 9843325 Ki = 4.22 nM T36059 C9M0GR 9843337 Ki = 4580 nM T36059 CKZ07C 9843424 Ki = 3162.28 nM T36059 C7HAP8 9843843 Ki > 10000 nM T36059 CDO4W1 9844103 Ki >> 10000 nM T36059 CZDJ43 9845174 Ki > 10 nM T36059 CXY6N1 9847046 Ki = 124 nM T36059 CRLO45 9850648 Ki = 1.5 nM T36059 C2F8KA 9850900 Ki = 284 nM T36059 CUB8T7 9857266 Ki = 1075 nM T36059 CUZL86 9857422 Ki = 136 nM T36059 CP50JH 9857698 Ki = 360 nM T36059 CUO04X 9857735 Ki = 302 nM T36059 CYXI30 9858577 Ki = 1779 nM T36059 C6IK1X 9858578 Ki = 2204 nM T36059 CUGV50 9860013 Ki = 476 nM T36059 CZRS26 9863617 Ki = 0.28 nM T36059 CH7AO5 9864945 Ki = 8.29 nM T36059 CTK0Z8 9865923 Ki = 73 nM T36059 CZN45Y 9865975 Ki = 112 nM T36059 CV19SJ 9868763 Ki = 40 nM T36059 CRJ04W 9868991 Ki = 55 nM T36059 C7ARK4 9870396 Ki = 54 nM T36059 CQR53Y 9870718 Ki = 61.9 nM T36059 CG47TN 9870719 Ki = 352 nM T36059 CQ4LC2 9872676 Ki = 628 nM T36059 CQ0T4V 9880392 Ki = 871 nM T36059 CYPJ74 9880921 Ki = 168 nM T36059 C5URA3 9881967 Ki = 18 nM T36059 CB26YS 9883190 Ki = 568 nM T36059 CZJV79 9885200 Ki = 2010 nM T36059 C67XMD 9885883 Ki = 2170 nM T36059 CZN50C 9887859 Ki = 0.01 nM T36059 CLIE16 9890003 Ki = 2.78 nM T36059 C7C5VN 9890439 Ki = 140 nM T36059 CY71UN 9892149 Ki = 121 nM T36059 CNAJ03 9892397 Ki = 109 nM T36059 C8LSD7 9893136 EC50 = 0.67 nM T36059 C0RCP7 9901171 Ki = 792 nM T36059 CDPV97 9901196 Ki = 491 nM T36059 CW8PY4 9901260 Ki = 440 nM T36059 CJKD76 9901497 Ki = 693 nM T36059 CW8Z9K 9901700 Ki = 563 nM T36059 CTU57Q 9902350 IC50 = 26 nM T36059 CA52RY 9902562 Ki = 338 nM T36059 CJ3OC1 9902563 Ki = 1256 nM T36059 C7YM0O 9904456 Ki = 35 nM T36059 CUG70S 9906178 Ki = 170 nM T36059 CQ3WL2 9909886 Ki = 59.9 nM T36059 CR4SN0 9910158 Ki = 1.6 nM T36059 C91GXW 9910620 Ki = 82.8 nM T36059 CDN1R5 9910926 Ki = 0.49 nM T36059 CC9FE0 9912816 Ki = 79.2 nM T36059 CO9WC2 9922606 Ki = 120 nM T36059 CMGL57 9923269 Ki = 1931 nM T36059 CO7FP5 9924271 Ki = 304 nM T36059 C8CU7X 9924272 Ki = 24 nM T36059 CO52VW 9924325 Ki = 16 nM T36059 CLK76N 9924994 Ki = 37 nM T36059 CXWU86 9929340 Ki = 2.1 nM T36059 C7X1TD 9929470 Ki = 0.16 nM T36059 C3H4WX 9930260 Ki = 15300 nM T36059 CPC4I6 9931686 Ki = 51.1 nM T36059 C8TMY5 9932840 Ki = 0.42 nM T36059 C3OU5G 9933719 Ki = 22.5 nM T36059 C9RYN2 9935097 Ki = 2640 nM T36059 CJ5YV8 9935943 Ki > 5000 nM T36059 CO3MX7 9935978 Ki = 14.8 nM T36059 CY82JD 9936058 Ki = 670 nM T36059 CR05XW 9936467 Ki = 363 nM T36059 CW4NR7 9945226 Ki = 269 nM T36059 CL3MY6 9946338 Ki = 220 nM T36059 CBZG96 9949541 Ki = 1472 nM T36059 C4MSO1 9950776 Ki > 1000 nM T36059 C9F7BL 9953799 Ki = 0.28 nM T36059 C2KD6M 9954747 Ki = 130 nM T36059 C8WR2V 9955052 Ki = 3.396 nM T36059 C4OG6P 9956774 Ki = 3250 nM T36059 C7GH6I 9957239 Ki = 922 nM T36059 CJUC15 9958472 Ki = 1.2 nM T36059 CPGT28 9967620 Ki = 844 nM T36059 C2UF7H 9968253 Ki = 1174 nM T36059 CDM42Y 9970296 Ki = 380 nM T36059 CMZ6X7 9970667 Ki > 10000 nM T36059 CVR5X8 9974009 Ki = 5 nM T36059 CZE6O5 9975036 Ki = 104 nM T36059 CZVI16 9976651 EC50 = 15848931.92 nM T36059 C2QYW9 9976989 Ki = 340 nM T36059 C5SZL7 9978117 Ki = 5 nM T36059 CLI90J 9981945 Ki = 23 nM T36059 CLZ2G0 9982930 Ki = 42.9 nM T36059 C5F1IV 9985321 Ki = 8 nM T36059 C06EVM 9995603 Ki = 96 nM T36059 CLN8X6 9996279 Ki = 0.6 nM T36059 CP0E1S 9996282 Ki = 9.6 nM T36059 CJ83TP 9999033 Ki = 790 nM T36059 CMP5T0 10007115 Ki = 300 nM T36059 C2TCR6 10007492 Ki = 44.3 nM T36059 C2WSC5 10014953 Ki = 0.79 nM T36059 CPAT84 10020580 Ki = 4.7 nM T36059 CA4X5Z 10026670 Ki > 10000 nM T36059 C9E4GW 10029879 Ki = 1300 nM T36059 CP2ZS6 10039961 Ki = 2.1 nM T36059 CJZY04 10040075 Ki = 47 nM T36059 CTQE97 10040914 Ki = 16 nM T36059 CH5J8G 10042508 Ki = 0.19 nM T36059 CL2KT4 10042766 Ki = 580000 nM T36059 CKD5L0 10043187 Ki = 55.4 nM T36059 CS5IX1 10045523 Ki = 44.9 nM T36059 CX32QD 10046002 Ki = 4.4 nM T36059 CLRM29 10046145 Ki > 10000 nM T36059 CZY7A5 10046345 Ki = 3.8 nM T36059 CU7EA4 10047690 Ki = 1.7 nM T36059 C3X1QT 10050031 Ki > 10000 nM T36059 C1I2LX 10062252 Ki > 10000 nM T36059 CX59SD 10062568 Ki = 78 nM T36059 CM39QU 10063481 Ki = 4219 nM T36059 CJW0D6 10063525 Ki = 257 nM T36059 C7EKU9 10063737 Ki = 3.4 nM T36059 CGE17I 10065148 Ki = 224 nM T36059 C7K3ID 10066439 Ki = 26 nM T36059 C0HBO3 10067267 Ki = 173 nM T36059 C6VLS0 10075248 Ki = 475 nM T36059 C1W0YH 10083550 Ki = 33 nM T36059 CQ7TL1 10084926 Ki = 788 nM T36059 C1LKV6 10085895 Ki = 91.4 nM T36059 C42KUZ 10108084 Ki = 6 nM T36059 CK4M6F 10114333 Ki = 160 nM T36059 C78NYU 10131882 IC50 = 45 nM T36059 C5WDR4 10132256 Ki = 124 nM T36059 C1AU0B 10150517 Ki = 270 nM T36059 CV87WF 10153029 IC50 = 1467 nM T36059 CZ17TE 10153190 Ki > 1000 nM T36059 C6IC0Y 10154604 Ki = 698 nM T36059 CBY63V 10155413 Ki = 736 nM T36059 C7OC0T 10156654 IC50 = 8.2 nM T36059 C7J5EN 10158974 Ki = 700 nM T36059 C4FNY6 10175278 Ki > 1000 nM T36059 C4GOP3 10180118 IC50 = 22 nM T36059 CUC8Y6 10196060 IC50 = 8888 nM T36059 C5NOP9 10196114 Ki > 167 nM T36059 C1NW4L 10196517 IC50 = 4314 nM T36059 CRY0O1 10200261 EC50 = 0.000001 nM T36059 C9KP1Y 10218183 IC50 = 5249 nM T36059 CN9W0F 10225178 Ki = 0.19 nM T36059 C84YAW 10237847 IC50 = 1315 nM T36059 CZE01H 10238677 IC50 = 844 nM T36059 CP7K3D 10246959 Ki = 2.03 nM T36059 C5RKX3 10247091 Ki = 650 nM T36059 CH7J2I 10248282 Ki = 74 nM T36059 C2HVY5 10248379 Ki = 15.85 nM T36059 CH7VN4 10249674 Ki > 10000 nM T36059 C0TXB5 10250190 Ki = 9830 nM T36059 C0CG8M 10253877 Ki = 2 nM T36059 CGMN21 10254700 Ki = 3.8 nM T36059 CT41UJ 10256007 Ki = 288 nM T36059 C9RSB2 10256116 Ki = 2.39 nM T36059 CS80UL 10257979 Ki = 7.413 nM T36059 CF1UN5 10267860 Ki = 1048 nM T36059 CA3S5M 10269139 IC50 = 35 nM T36059 CB5DN6 10288169 IC50 = 2085 nM T36059 CH6ZC0 10288197 IC50 = 1525 nM T36059 CI5LZ3 10291235 Ki = 11 nM T36059 C0VY4L 10291948 Ki = 10 nM T36059 C8RM9P 10292899 EC50 = 794328.23 nM T36059 C40WZO 10296638 Ki = 0.14 nM T36059 CI2E8K 10308937 Ki = 120 nM T36059 CU17KP 10310578 IC50 = 6438 nM T36059 C8BO9X 10310768 Ki > 9000 nM T36059 CC21BD 10311222 IC50 = 3169 nM T36059 CBSE14 10311510 Ki = 5 nM T36059 C0H5MU 10316176 Ki = 76.7 nM T36059 CXY40F 10318983 Ki > 10000 nM T36059 C4MPT3 10324445 Ki = 8.58 nM T36059 CUBQ81 10334707 Ki = 44.1 nM T36059 CR9HV2 10338742 Ki = 2560 nM T36059 CO24NY 10338801 Ki = 2 nM T36059 CF5N9O 10339165 Ki = 80.8 nM T36059 CZ81IA 10342970 Ki = 3.7 nM T36059 C0XHI4 10345159 Ki = 1250 nM T36059 C5Y1NM 10345700 Ki = 610 nM T36059 CTR36D 10345757 Ki = 4.2 nM T36059 C7IPE9 10346511 Ki = 0.22 nM T36059 CD7C2A 10359522 Ki = 4 nM T36059 CAW15E 10359831 Ki = 96 nM T36059 CLH34K 10361707 Ki = 31 nM T36059 C1RFV6 10362099 Ki > 10000 nM T36059 C2R9YK 10369458 Ki = 29 nM T36059 CHZ32J 10377463 Ki = 331.13 nM T36059 C2PNT5 10380218 Ki = 126 nM T36059 C5HPZ3 10387088 Ki = 90.3 nM T36059 C73CUW 10387599 Ki = 697 nM T36059 CUP34N 10388920 Ki = 3.9 nM T36059 CR53SP 10390495 Ki = 0.87 nM T36059 C5F4WP 10403711 Ki = 108 nM T36059 C4UX5I 10404217 Ki = 4622 nM T36059 CA30OM 10406540 Ki > 10000 nM T36059 CZ1N7V 10407390 Ki = 222 nM T36059 CN1A2W 10407895 Ki = 128 nM T36059 C6YMN7 10415270 Ki = 7.8 nM T36059 C4LMK8 10421804 Ki = 2098 nM T36059 CO95VK 10422626 Ki = 70.8 nM T36059 CAJ68I 10426659 Ki = 786 nM T36059 CWUB34 10431614 Ki = 0.2897 nM T36059 C9D5ZQ 10431643 Ki = 814 nM T36059 CNO9Z0 10436397 Ki = 3.3 nM T36059 CO4H0C 10436433 Ki = 130 nM T36059 CXOL94 10438449 IC50 = 6700 nM T36059 C6BH4D 10449090 Ki = 25.8 nM T36059 CSD86M 10449535 Ki = 23 nM T36059 C8XFL5 10449783 Ki > 10000 nM T36059 CZ9VB4 10450691 Ki = 2.2 nM T36059 C1BW6K 10451086 Ki = 27.5 nM T36059 C9FQ6C 10452788 Ki = 422 nM T36059 CK9FA7 10453097 Ki = 0.3396 nM T36059 CM4C2X 10455080 Ki = 0.2 nM T36059 CGM46Y 10455852 Ki = 1.5 nM T36059 C4OMF3 10468228 Ki = 2 nM T36059 C15VAO 10471588 Ki = 2.9 nM T36059 CI3LE9 10471721 Ki = 60.5 nM T36059 C5Y6IP 10472803 Ki = 4.2 nM T36059 CJ0U1M 10474279 Ki = 244 nM T36059 CT5RM2 10481541 Ki = 219 nM T36059 CQ1JW6 10481542 Ki = 219 nM T36059 C8RA6W 10482029 Ki = 2.3 nM T36059 CBGS14 10492556 Ki = 3600 nM T36059 CM40PW 10499201 Ki = 1700 nM T36059 CT9A5L 10499931 Ki = 108 nM T36059 CKA37B 10501538 Ki = 1100 nM T36059 CZ1J3U 10503669 Ki = 570 nM T36059 CO97UP 10505508 Ki = 33.8 nM T36059 CHC23X 10505816 Ki = 19.81 nM T36059 CGK7S5 10506248 Ki = 286 nM T36059 CSJN79 10506635 Ki = 436 nM T36059 CG1WL9 10514262 Ki = 600 nM T36059 C3IY7X 10517992 Ki = 2.9 nM T36059 CT4E5Q 10518459 Ki = 48.2 nM T36059 C8LZ0C 10520259 Ki = 4470 nM T36059 CA6L2E 10522079 Ki = 115000 nM T36059 C9OJF7 10522801 Ki = 32.9 nM T36059 C84SGE 10525928 Ki = 169 nM T36059 C5AY6C 10526022 Ki = 31.1 nM T36059 CFO9I6 10527314 Ki > 100000 nM T36059 C08OQV 10528161 Ki > 10000 nM T36059 CZ4JQ0 10528906 Ki = 3200000 nM T36059 CD78AR 10538513 Ki = 20000000 nM T36059 CFOS68 10539663 Ki > 10000 nM T36059 C5ATC3 10541585 Ki = 28.5 nM T36059 C9A0YD 10544617 Ki = 15.8 nM T36059 CA8P6H 10547577 Ki = 2128 nM T36059 CSOX08 10549896 Ki = 28.9 nM T36059 C6I8ML 10550526 Ki = 230000 nM T36059 C6I2PQ 10551147 Ki = 27.7 nM T36059 C82JRX 10551807 Ki = 1020 nM T36059 C68TYK 10551919 Ki = 2580 nM T36059 CN26SH 10551960 Ki = 520 nM T36059 CL10FM 10551961 Ki = 650 nM T36059 COL8H0 10552207 Ki = 3850 nM T36059 CTJF92 10552717 Ki = 0.586 nM T36059 C19LKF 10553234 Ki = 194 nM T36059 C53QCT 10554064 Ki = 240 nM T36059 C8RJI2 10554473 Ki = 2020 nM T36059 CTR56S 10564520 Ki = 80 nM T36059 C3C8WE 10565773 Ki = 309 nM T36059 CON7B0 10566365 Ki = 1900 nM T36059 CZ90RO 10566417 Ki = 8700 nM T36059 CC84VI 10567830 Ki = 420 nM T36059 CO34PZ 10568317 Ki = 1813 nM T36059 CIT8M6 10569148 Ki = 287000 nM T36059 CZ9PS2 10569216 Ki = 210 nM T36059 CZ7W5I 10569328 Ki = 22.3 nM T36059 CVW26Q 10570266 Ki = 44.1 nM T36059 CE3US5 10571608 Ki = 56.5 nM T36059 CVBD40 10572142 Ki = 310 nM T36059 C2T8YC 10572535 Ki > 10000 nM T36059 C1T3GL 10573122 Ki = 159 nM T36059 CH4ND1 10573130 Ki = 262 nM T36059 C16QBJ 10573891 Ki = 2800 nM T36059 C39ASY 10573999 Ki = 23 nM T36059 CBZ09J 10574014 Ki = 23.6 nM T36059 C2S8TH 10577289 Ki = 57.9 nM T36059 CRSD46 10577428 Ki = 44.7 nM T36059 C1E9AJ 10578123 Ki = 62.9 nM T36059 CL23DC 10580789 Ki = 25 nM T36059 CEW4T3 10587109 Ki = 299.92 nM T36059 CKI69M 10588725 Ki = 45.3 nM T36059 CIY5W3 10591699 Ki = 9180 nM T36059 CI6GS7 10594353 Ki = 27 nM T36059 C5Z4WV 10594397 Ki = 14.6 nM T36059 CVC8Y5 10596858 Ki = 40.9 nM T36059 C1P5DO 10597086 Ki = 81.3 nM T36059 CQ7S4X 10600124 Ki = 58.5 nM T36059 C02GZY 10601859 Ki = 42.65 nM T36059 CXM9I7 10602212 Ki = 346 nM T36059 C5W4XH 10602268 Ki > 10000 nM T36059 CY59KG 10602509 Ki = 1410 nM T36059 CS2VT6 10605011 Ki = 70.96 nM T36059 C34GYL 10613570 Ki = 8170 nM T36059 CSO52M 10613752 Ki = 150 nM T36059 C6M1NH 10613770 Ki = 157 nM T36059 CCU6M1 10615431 Ki = 1700 nM T36059 CQ1UA4 10615661 Ki = 78700000 nM T36059 C2N5UX 10616023 Ki = 2100 nM T36059 CLH03M 10616222 Ki = 13.9 nM T36059 C2VHD3 10616645 Ki = 82 nM T36059 CL8WG1 10617844 Ki = 35.8 nM T36059 CR1O9S 10617992 Ki = 54.6 nM T36059 C2T5LI 10618263 Ki = 115 nM T36059 CQ8X5N 10618368 Ki = 45500 nM T36059 CO2W4F 10619508 Ki = 1860 nM T36059 CGMH35 10619822 Ki = 1.47 nM T36059 CD57YJ 10620261 Ki = 2090 nM T36059 CD52HB 10620597 Ki = 193 nM T36059 C9X2UW 10621792 Ki = 647 nM T36059 C5JAK7 10621898 Ki = 0.362 nM T36059 CPLR23 10621961 Ki = 3.56 nM T36059 C0QI7Y 10622356 Ki = 2640 nM T36059 C8JB3I 10623248 Ki = 0.3199 nM T36059 CG4NS5 10624745 Ki = 22 nM T36059 CY6QP1 10626463 Ki = 51 nM T36059 CTS9Z3 10637031 Ki = 16000 nM T36059 C3INO8 10637656 Ki = 63 nM T36059 C7QWO6 10637742 Ki = 599.79 nM T36059 C9NKW1 10638807 Ki = 329 nM T36059 C2RTK9 10639706 Ki = 660 nM T36059 C78YHS 10641040 Ki > 10000 nM T36059 CP86LA 10641062 Ki = 152 nM T36059 C7LN3U 10642208 Ki = 506 nM T36059 CNQ5H4 10642873 Ki = 21.5 nM T36059 C5FY9Z 10642901 Ki = 1260000 nM T36059 CWKH90 10645626 Ki = 3130 nM T36059 C8O4LD 10645750 Ki > 10000 nM T36059 CD78NU 10646456 Ki = 14.4 nM T36059 C8O2UT 10647227 Ki = 0.5998 nM T36059 CFYN54 10647445 Ki = 59 nM T36059 C05SPI 10649436 Ki = 213 nM T36059 CKQ8P1 10649879 Ki = 882 nM T36059 C24IYH 10650201 Ki = 49.3 nM T36059 CBI7X5 10659581 Ki = 331 nM T36059 CZ97XY 10661229 Ki = 3.2 nM T36059 C8H1QL 10661355 Ki = 340 nM T36059 C8NCG3 10661707 Ki = 1148.15 nM T36059 C29LYV 10663485 Ki = 1246 nM T36059 CQ26WN 10664934 Ki = 336000 nM T36059 C0U2LA 10665761 Ki = 330 nM T36059 C2MN3W 10665887 Ki = 23900 nM T36059 CVIR83 10667072 Ki = 548 nM T36059 CHQ6B9 10668865 Ki > 10000 nM T36059 CCT9Y2 10669560 Ki = 72.1 nM T36059 CWTP16 10672116 Ki = 10900 nM T36059 CQ80BN 10673341 Ki = 53.7 nM T36059 CL3ZF5 10674624 Ki = 465 nM T36059 CI87XU 10686088 Ki = 504 nM T36059 CG8W6T 10687044 Ki = 117000 nM T36059 CGU6W0 10687707 Ki > 10000 nM T36059 CMI92Q 10688603 Ki = 180 nM T36059 C5RMA3 10688700 Ki = 322 nM T36059 C6SV1Y 10689930 Ki > 10000 nM T36059 C8FDB3 10690524 Ki = 87300 nM T36059 CQV6Y1 10691504 Ki = 82.5 nM T36059 CZ6E4D 10695619 Ki = 856 nM T36059 CHLI76 10696384 Ki = 446 nM T36059 C9B1PF 10696675 Ki = 7.998 nM T36059 CNO6X0 10696777 Ki = 188 nM T36059 CW4Q7M 10697195 Ki = 243 nM T36059 CVXR28 10697531 Ki = 364 nM T36059 CC0G1W 10709706 Ki = 800 nM T36059 C5EM0D 10709852 Ki = 45 nM T36059 CO0WC9 10710278 Ki = 114 nM T36059 CPV34D 10711231 Ki = 147000 nM T36059 C13OJI 10714291 Ki = 194 nM T36059 C92JZT 10719181 Ki = 1200 nM T36059 CFT53W 10719352 Ki = 220 nM T36059 C07JSG 10720065 Ki = 1862.09 nM T36059 CS41HM 10720163 Ki = 379 nM T36059 CBFG43 10720641 Ki = 23.8 nM T36059 CVI9S1 10722996 Ki = 1250 nM T36059 CKMJ53 10732242 Ki = 90.2 nM T36059 CTR6Z8 10732372 Ki = 36.6 nM T36059 C9IJL3 10734376 Ki = 2 nM T36059 C9PRY0 10735167 Ki = 257000 nM T36059 CD2AF5 10735584 Ki = 8500 nM T36059 C3K7FG 10735745 Ki = 1990 nM T36059 CE3G2Z 10736931 Ki = 248 nM T36059 C7NXS3 10737168 Ki = 429.54 nM T36059 C8YU9P 10738970 Ki = 188 nM T36059 CWX81Q 10741090 Ki = 960 nM T36059 CHP9A0 10744813 Ki = 170000 nM T36059 CBHU92 10745030 Ki = 1350 nM T36059 CB0L1T 10745111 Ki = 16 nM T36059 C2S0OJ 10746790 Ki = 348 nM T36059 C03CBY 10755990 Ki = 48.3 nM T36059 CFWH27 10756111 Ki = 3600 nM T36059 C82ZXO 10758495 Ki = 3300 nM T36059 CG67NI 10759742 Ki = 707 nM T36059 CVM5F2 10760994 Ki = 155 nM T36059 CWK2M9 10761106 Ki = 700 nM T36059 CUEK94 10761731 Ki = 4 nM T36059 CXBH30 10761984 Ki = 220000 nM T36059 CTED21 10762042 Ki = 42.5 nM T36059 C1XB8G 10762204 Ki = 9.9 nM T36059 C5D8YL 10763173 Ki = 56.1 nM T36059 C7LN1B 10764269 Ki = 4830 nM T36059 CCZ4U8 10765059 Ki = 0.4797 nM T36059 CO4XR0 10766011 Ki > 10000 nM T36059 CL6VU1 10766773 Ki = 874 nM T36059 CK0C8P 10767043 Ki = 391 nM T36059 C0FVU4 10767601 Ki = 65 nM T36059 C7ZJL6 10768474 Ki = 17.5 nM T36059 CR23JY 10768475 Ki = 577 nM T36059 C5B6KP 10769581 Ki = 4481 nM T36059 CIRS48 10778887 Ki = 490 nM T36059 CN3AC0 10778962 Ki = 197 nM T36059 C3GJ5Z 10779327 IC50 = 40.2 nM T36059 CF1V9Q 10783420 Ki = 670 nM T36059 CNC32V 10785815 Ki = 44.2 nM T36059 CPBH31 10788003 Ki = 211 nM T36059 CW5N4X 10789143 Ki = 32.1 nM T36059 C79MNZ 10791347 Ki = 0.98 nM T36059 CYG2J5 10792296 Ki = 213 nM T36059 CM1N7O 10793100 Ki = 36 nM T36059 C3SCU6 10802472 Ki = 404 nM T36059 C53GTE 10803557 Ki = 25 nM T36059 C7Y8EJ 10803880 Ki = 4000 nM T36059 CH1A3F 10804397 Ki = 68.4 nM T36059 CMB81D 10808093 Ki = 1200 nM T36059 CJ1E7A 10809682 Ki = 1870 nM T36059 CH5U3A 10810142 Ki = 5580 nM T36059 CU6G3T 10810590 Ki = 137 nM T36059 CMBR87 10811905 Ki = 9.67 nM T36059 C2N5AB 10812872 Ki > 10000 nM T36059 C47WZO 10813707 Ki = 6.71 nM T36059 CF81JV 10813915 Ki = 109 nM T36059 CD97KF 10814245 Ki = 1140 nM T36059 CE39PU 10816300 Ki = 46.3 nM T36059 CXV35E 10817403 Ki = 538 nM T36059 C7BT0O 10824674 Ki > 10000 nM T36059 CS7YB8 10826246 Ki = 79.2 nM T36059 C4ZX9L 10826247 Ki = 118 nM T36059 CM0S5H 10827471 Ki = 91 nM T36059 CB1X3E 10828275 Ki = 10000 nM T36059 C1N0QG 10829180 Ki = 479 nM T36059 CHZK51 10830023 Ki = 137 nM T36059 C7XJ0O 10831497 Ki > 10000 nM T36059 CT1RA3 10832042 Ki = 264000 nM T36059 CCUG91 10832101 Ki = 150000 nM T36059 CD10KA 10832948 Ki = 2040000 nM T36059 CR8G2F 10834400 Ki = 8.3 nM T36059 C6Q2MG 10834512 Ki = 3.75 nM T36059 C6UP5K 10834513 Ki = 3416 nM T36059 CCB9N0 10834552 Ki = 276 nM T36059 C7PHL9 10834790 Ki = 55.1 nM T36059 CF2R3V 10837382 Ki = 2410 nM T36059 CBN26U 10837543 Ki = 46.3 nM T36059 CPLT60 10838118 Ki = 32.9 nM T36059 C0KIA2 10838283 Ki = 2750 nM T36059 C2E6PX 10839228 Ki = 31 nM T36059 C20WTU 10839296 Ki = 138 nM T36059 C4H7NS 10839874 Ki = 483 nM T36059 C89OKC 10840167 Ki = 2300 nM T36059 CD4C9P 10849846 Ki = 354 nM T36059 C6CSZ4 10852375 Ki = 81 nM T36059 CE04SL 10852506 Ki = 699.84 nM T36059 C1CM2Q 10853502 Ki = 580 nM T36059 C25DVO 10854498 Ki = 370000 nM T36059 C4BWE6 10854560 Ki = 940 nM T36059 C3I2WZ 10859484 Ki = 225 nM T36059 CSH1O4 10859911 Ki = 202 nM T36059 C3QWZ1 10862463 Ki = 17 nM T36059 CZ7WJ9 10863425 Ki = 2.999 nM T36059 CRU6I1 10863910 Ki = 676 nM T36059 C4J8CR 10868826 Ki = 3850 nM T36059 CJ5G9S 10870151 Ki = 23.3 nM T36059 C7RD3K 10872091 Ki > 10000 nM T36059 CKE05V 10872482 Ki = 104 nM T36059 C4HO6X 10874051 Ki = 212 nM T36059 CWL1K9 10874724 IC50 = 3730 nM T36059 CB6J8X 10875138 Ki = 102 nM T36059 C2B1MG 10878835 Ki = 2000 nM T36059 C47HSO 10882425 Ki = 2857 nM T36059 C1AL7H 10884000 Ki > 1000 nM T36059 CCV1Q4 10884004 Ki = 88.3 nM T36059 CN8J0Y 10884265 Ki = 0.2399 nM T36059 CY62BK 10884803 Ki = 0.8091 nM T36059 CRI50E 10885636 IC50 = 3480 nM T36059 C9YZ3M 10885937 Ki = 1.6 nM T36059 CP0M3N 10892251 Ki = 3050 nM T36059 CLGC13 10893465 Ki = 17.4 nM T36059 CIG9Z2 10895416 Ki = 0.3396 nM T36059 C2P1QB 10895565 Ki = 50 nM T36059 CU5KZ3 10896741 Ki = 7.3 nM T36059 C6FH3A 10896988 Ki = 20.5 nM T36059 C42SFP 10904208 Ki = 79 nM T36059 C2LV6K 10904370 Ki > 1000 nM T36059 C3BGR7 10904704 Ki > 1000 nM T36059 CU93CT 10904839 Ki > 10000 nM T36059 C3KOX6 10905184 Ki = 0.31 nM T36059 CKV30L 10905799 Ki = 0.21 nM T36059 CH52LS 10906943 Ki = 215 nM T36059 CX65PW 10907460 IC50 = 2460 nM T36059 C0D8YH 10907478 Ki = 9.1 nM T36059 C4H8PS 10914466 Ki = 3 nM T36059 CI87AW 10915653 Ki = 110 nM T36059 CJ52TM 10916451 Ki > 10000 nM T36059 CS58FH 10917575 Ki = 110 nM T36059 CVFL61 10918042 Ki = 0.9099 nM T36059 CGXE04 10925715 Ki = 20.2 nM T36059 CQXA29 10926253 Ki > 1000 nM T36059 CCO41S 10926422 Ki = 80.6 nM T36059 C3IA5Y 10927361 Ki = 13660 nM T36059 CJB64E 10927693 Ki = 0.9099 nM T36059 CFZ49H 10928011 Ki > 10000 nM T36059 C1B6XL 10928182 Ki = 0.3396 nM T36059 CG2N7W 10928649 Ki = 0.5495 nM T36059 C7F8YE 10937272 Ki = 526 nM T36059 C58CRE 10938276 Ki = 0.14 nM T36059 CG24MW 10938325 Ki > 10000 nM T36059 C6FQ3L 10938608 Ki = 0.3999 nM T36059 CM0OS2 10939174 IC50 = 5470 nM T36059 C8BLN4 10939224 Ki = 0.2999 nM T36059 C2BPD4 10949114 Ki = 114 nM T36059 CSE18R 10958838 Ki = 5800 nM T36059 CXWV50 10959335 Ki > 10000 nM T36059 CY2OS9 10961304 Ki = 14 nM T36059 C7YVC5 10962009 Ki > 10000 nM T36059 CAM58P 10968439 Ki > 10000 nM T36059 CXH12M 10970127 Ki = 173 nM T36059 CD4MO1 10970525 Ki = 1184 nM T36059 CLK8M1 10970782 Ki > 10000 nM T36059 CKE84F 10970819 Ki = 2.3 nM T36059 C7TUS2 10970979 Ki = 77 nM T36059 CD16UB 10971099 Ki = 1.03 nM T36059 C9WLT0 10971427 Ki > 10000 nM T36059 C6OFK0 10971806 Ki = 0.859 nM T36059 C4ZU8F 10971841 Ki = 0.2897 nM T36059 CBW9J6 10972594 Ki > 10000 nM T36059 C8F9LD 10979983 Ki > 10000 nM T36059 C2TEB7 10981207 Ki = 1192 nM T36059 CZ57WA 10981863 Ki = 2320 nM T36059 C4G0YQ 10982985 Ki = 0.7096 nM T36059 CO5PH3 10984232 Ki = 1100 nM T36059 C83XMH 10993869 Ki > 10000 nM T36059 C6BH4T 10993916 Ki = 0.7396 nM T36059 C9NP1R 10994142 Ki > 1000 nM T36059 C3F4TJ 10994183 Ki = 0.5 nM T36059 CSO19C 10994216 Ki = 5.49 nM T36059 C31HJV 10994317 Ki = 0.51 nM T36059 CH6Y5I 11000858 Ki = 2250 nM T36059 C9IGK2 11003653 Ki = 10000 nM T36059 CR67WG 11003842 Ki = 67 nM T36059 CJ6C9K 11003971 IC50 = 3330 nM T36059 CMDB43 11004373 Ki = 0.2999 nM T36059 C8CS2Y 11004885 Ki = 558 nM T36059 CEP35L 11004986 Ki > 1000 nM T36059 CLR4B8 11005067 Ki > 10000 nM T36059 CJC9K4 11005810 IC50 = 5980 nM T36059 C2QJW7 11013957 Ki = 8.3 nM T36059 C0KDE3 11014188 Ki = 0.8091 nM T36059 C47IDH 11014608 Ki = 9.7 nM T36059 C6EQD3 11015003 Ki = 0.859 nM T36059 C30WTZ 11017082 Ki > 10000 nM T36059 CI3E7D 11019436 Ki > 100000 nM T36059 C9TPE8 11022827 Ki = 580 nM T36059 C20KVX 11025671 Ki = 253 nM T36059 C8UPZ3 11026001 Ki = 0.53 nM T36059 CF5B8Z 11026358 Ki > 1000 nM T36059 CPD61T 11026434 Ki = 0.65 nM T36059 C12YXH 11027282 Ki > 10000 nM T36059 CX28EA 11027412 Ki = 40 nM T36059 CPV27K 11027743 Ki = 24 nM T36059 CW05DS 11028588 Ki > 1000 nM T36059 C5I8UZ 11035880 Ki = 3.162 nM T36059 CA2QL9 11036560 Ki = 1125 nM T36059 CHEA89 11037671 Ki > 10000 nM T36059 CR7FM2 11037739 Ki = 0.4295 nM T36059 CM9FK6 11037972 Ki = 0.3698 nM T36059 CE0YZ4 11038875 Ki = 7.4 nM T36059 CPB50W 11045730 Ki = 40 nM T36059 C50MFV 11046203 Ki = 477 nM T36059 CUV0P9 11046285 Ki = 6.3 nM T36059 C4HDC2 11046837 Ki = 200 nM T36059 C85NWI 11047444 Ki = 32.3 nM T36059 C23JHR 11047568 IC50 = 4180 nM T36059 CVQ3B8 11047906 Ki = 213 nM T36059 CS8P0U 11048163 Ki > 10000 nM T36059 CL1RP8 11048438 Ki = 4.9 nM T36059 C6EBF3 11048769 IC50 = 1510 nM T36059 CW7Q6U 11053743 Ki = 5780 nM T36059 CL29NE 11056301 Ki = 36 nM T36059 CTZM01 11058084 Ki = 1240 nM T36059 CCS8A6 11058550 Ki = 0.6998 nM T36059 CFJG64 11059058 IC50 = 1780 nM T36059 CYZ83I 11059351 Ki = 0.57 nM T36059 CA91IB 11060260 Ki > 10000 nM T36059 CM7TR4 11068963 Ki = 3.388 nM T36059 C9KRQ1 11070905 Ki = 30 nM T36059 CG41BK 11071079 IC50 = 4210 nM T36059 C81MOC 11071091 IC50 = 3750 nM T36059 C7HIP2 11071159 Ki > 1000 nM T36059 C0QM4E 11078375 Ki = 26.7 nM T36059 CN5S7E 11078951 Ki = 308 nM T36059 C1EJI0 11080491 Ki = 81 nM T36059 CKX4G6 11080788 Ki = 0.5998 nM T36059 C4Y7NZ 11081189 Ki = 2.5 nM T36059 CV9Q3D 11088133 Ki = 33.3 nM T36059 CKEF14 11089092 Ki = 1217 nM T36059 C83TJN 11090423 Ki = 950 nM T36059 CR3X1M 11091600 Ki > 1000 nM T36059 C64PWO 11091632 Ki = 0.859 nM T36059 C15EQZ 11091783 Ki = 183 nM T36059 CZW34N 11099564 Ki = 14 nM T36059 CVDM13 11102838 Ki > 1000 nM T36059 C0DXW3 11109201 Ki > 10000 nM T36059 CMY97P 11112381 Ki = 1.2 nM T36059 C3Z5PU 11112543 Ki = 0.5598 nM T36059 CJ21DZ 11112670 Ki = 409 nM T36059 C6RB5D 11112711 Ki = 1.4 nM T36059 C3IFX4 11112849 Ki = 0.2698 nM T36059 C7DE0U 11113605 IC50 = 5080 nM T36059 CBFQ96 11121771 Ki = 1119 nM T36059 C9FGQ0 11122039 Ki = 32.3 nM T36059 CR7X2T 11122708 Ki = 0.2 nM T36059 CLN23H 11123135 Ki > 1000 nM T36059 C06JLD 11123887 Ki = 47 nM T36059 C4CWA8 11133107 Ki = 348 nM T36059 CJ86ZM 11133545 Ki = 0.4295 nM T36059 CL19OW 11133804 Ki = 0.3999 nM T36059 CTG5Y7 11133843 Ki = 0.7998 nM T36059 CTWX69 11141317 Ki = 45.6 nM T36059 CE04DU 11142587 Ki = 68 nM T36059 CH4TG2 11144119 Ki > 1000 nM T36059 C9N1RL 11144868 Ki = 0.46 nM T36059 C72QCG 11145314 Ki > 10000 nM T36059 C4AR0D 11150120 Ki = 91.2 nM T36059 CVF8Z5 11151115 IC50 = 12 nM T36059 C79YSE 11153187 Ki = 99 nM T36059 CX7WT4 11154027 Ki = 420 nM T36059 CLQR16 11157262 Ki = 83 nM T36059 C1FVD5 11162618 Ki = 1526 nM T36059 C7PEC2 11163042 Ki = 175 nM T36059 CNY65E 11163483 Ki = 11.2 nM T36059 CS0N2C 11164346 Ki = 24 nM T36059 C9P3VW 11164926 Ki = 1170 nM T36059 CJN5M3 11168952 Ki = 480 nM T36059 CPB62L 11174953 Ki = 171 nM T36059 C12UTW 11175566 Ki = 15 nM T36059 CU96ZO 11176782 Ki = 45 nM T36059 CJ02LB 11178828 Ki = 41 nM T36059 CE3TB0 11186762 Ki = 1720 nM T36059 CHD65Q 11198201 Ki > 1000 nM T36059 C2Y7RN 11199559 Ki = 670 nM T36059 CP14DE 11202227 Ki = 5.94 nM T36059 COW67H 11203547 Ki = 6.95 nM T36059 C41PYH 11209919 Ki = 0.8 nM T36059 C6JD3L 11210192 Ki = 96.2 nM T36059 CV5BC1 11211172 Ki = 1390 nM T36059 CUD65V 11213917 Ki = 4.48 nM T36059 CV5Y6A 11214123 Ki = 23 nM T36059 CQ0D6R 11214486 Ki = 11.89 nM T36059 CJ0E7L 11215089 Ki = 9.97 nM T36059 C3FP0D 11229946 Ki = 4670 nM T36059 C3B4ZF 11232994 Ki = 960 nM T36059 CRPX67 11233074 Ki = 1530 nM T36059 C9IHT1 11233411 Ki = 3.45 nM T36059 CB6Y4A 11233413 Ki = 125 nM T36059 CODS67 11233881 Ki = 1810 nM T36059 C4OB6K 11236128 Ki = 7.41 nM T36059 C1KM3O 11244144 Ki = 203 nM T36059 C57WSV 11244376 Ki = 178 nM T36059 CHD2E3 11248230 Ki = 6.699 nM T36059 CG0OL1 11254831 Ki = 335 nM T36059 CA4EP9 11255271 Ki = 49.8 nM T36059 C7LS3R 11256992 Ki = 74 nM T36059 CCU71Z 11257069 Ki = 60 nM T36059 CL1J5B 11257336 Ki ~ 10000 nM T36059 C86XNQ 11260448 Ki = 400 nM T36059 CK7SM8 11266431 Ki = 97 nM T36059 C90UAN 11267262 Ki = 83 nM T36059 CWGM03 11282593 Ki = 0.82 nM T36059 CGR1A8 11289861 Ki = 1483 nM T36059 C48JAP 11290020 Ki = 676 nM T36059 C8B2RV 11290216 Ki = 22 nM T36059 CW9GN1 11292054 Ki = 5400 nM T36059 CX17GU 11293096 Ki = 2770 nM T36059 CLW5H2 11301432 Ki = 382.5 nM T36059 C1KJC2 11301673 Ki = 429 nM T36059 CQ7O1I 11302588 Ki = 70 nM T36059 C4PH8A 11306173 Ki = 413 nM T36059 CUS2N9 11313850 Ki > 1000 nM T36059 CX7QW0 11324734 Ki = 70 nM T36059 CY8KX5 11329375 Ki = 1.5 nM T36059 CGCJ09 11335341 Ki = 73.2 nM T36059 CJX89P 11348709 Ki = 36 nM T36059 CEU9X7 11348760 Ki = 4.7 nM T36059 C3TH4B 11352497 Ki = 140 nM T36059 CEI47X 11353406 Ki = 1200 nM T36059 C2Z8GE 11358739 Ki = 176 nM T36059 CRND96 11360082 Ki = 80 nM T36059 C8G3FO 11371101 Ki = 8 nM T36059 CUF53H 11373346 Ki = 1700 nM T36059 CNPM32 11374351 Ki = 3.98 nM T36059 C6WGI3 11375013 Ki = 16.29 nM T36059 C0M8KH 11380777 Ki = 86.5 nM T36059 CB3J6T 11380878 Ki = 6437 nM T36059 CRU3A7 11381738 Ki = 1102 nM T36059 CSD31L 11386134 Ki > 10000 nM T36059 C8KD6J 11386951 Ki = 400 nM T36059 C21UDI 11387030 Ki = 2700 nM T36059 CB2C4P 11392671 Ki = 586 nM T36059 CVAJ46 11393155 Ki = 402 nM T36059 CXPM05 11394389 Ki = 23 nM T36059 CD8G3K 11405982 Ki = 1.95 nM T36059 C8AON6 11407615 Ki = 8.09 nM T36059 C6IVY0 11408692 Ki = 0.763 nM T36059 CLM04X 11412911 Ki > 1000 nM T36059 CLD1X7 11420910 Ki = 4300 nM T36059 CDVM74 11424338 Ki = 437 nM T36059 C30ZXP 11426423 Ki = 1390 nM T36059 CM5C6V 11427243 Ki = 100 nM T36059 CQ7H6Z 11427378 Ki = 39.6 nM T36059 CPS9L6 11427880 Ki = 170 nM T36059 CF4H1A 11428535 Ki = 31 nM T36059 C85LYP 11430418 IC50 > 1000 nM T36059 C1U0CT 11431149 Ki = 4.03 nM T36059 CL0W7H 11442248 Ki = 15 nM T36059 C65KVC 11451201 Ki = 2420 nM T36059 CY95OG 11451820 Ki = 1.009 nM T36059 C6CV1B 11452333 Ki = 115 nM T36059 C70ZYC 11454117 Ki = 7.83 nM T36059 CA6YD2 11461202 Ki = 25 nM T36059 CZIN71 11462033 Ki = 170 nM T36059 C5M3SD 11463674 Ki = 200 nM T36059 C5JTD0 11464552 Ki = 55 nM T36059 C9CFK5 11465677 Ki > 1000 nM T36059 C9NP2C 11466670 Ki = 1200 nM T36059 C9RK6X 11475577 Ki = 22 nM T36059 C83XMS 11475769 Ki = 2 nM T36059 C6CMF0 11478510 Ki = 5780 nM T36059 CE7JS1 11483771 Ki = 335 nM T36059 CFQJ87 11484984 Ki = 2050 nM T36059 CKNU87 11486094 Ki = 116 nM T36059 CNDF82 11487397 Ki = 20.53 nM T36059 C2SY3I 11492651 Ki = 3670 nM T36059 CI4JC0 11492857 Ki = 280 nM T36059 CF41GK 11493648 Ki = 28.2 nM T36059 CKN80I 11494063 Ki = 99 nM T36059 C5LN1D 11497238 Ki = 5.3 nM T36059 C3YG6W 11500266 Ki = 278 nM T36059 CK8Z4J 11501636 Ki = 1500 nM T36059 C6KL3S 11501678 Ki = 0.35 nM T36059 CUQ4Y9 11504806 Ki = 415 nM T36059 CQ97HE 11505814 Ki = 354 nM T36059 C0WV8M 11507345 Ki = 370 nM T36059 COG79X 11508049 Ki = 707 nM T36059 C0AWD8 11508923 Ki = 282 nM T36059 CI98OZ 11511703 Ki = 44 nM T36059 C8GL1J 11511804 Ki = 14 nM T36059 CA7PE0 11514585 Ki = 108 nM T36059 CH03ZF 11516748 Ki = 3.5 nM T36059 CN2DI8 11516857 Ki = 1.1 nM T36059 CD29AZ 11517013 Ki = 34 nM T36059 CN65IW 11521902 Ki = 420 nM T36059 CT60SW 11522152 Ki = 5880 nM T36059 CQNA38 11522379 Ki = 2.5 nM T36059 CS1M7B 11522670 Ki = 1850 nM T36059 CQZ37L 11524264 Ki = 5.1 nM T36059 CC23GO 11524705 Ki = 1 nM T36059 C1CJ2S 11525283 Ki >= 10000 nM T36059 CF2T1V 11526947 Ki = 342 nM T36059 CBZ5X2 11527814 Ki = 343 nM T36059 C21IUQ 11529194 Ki > 1000 nM T36059 CKC6F5 11529450 Ki = 84 nM T36059 CV2DP6 11530256 Ki = 1190 nM T36059 C6Z0EX 11531100 Ki = 138 nM T36059 C47MXO 11531253 Ki >= 10000 nM T36059 C46UMB 11531355 Ki = 22 nM T36059 CVY83E 11531978 Ki = 100 nM T36059 C92FYA 11533614 EC50 = 1640 nM T36059 C19JCF 11533636 Ki = 3.29 nM T36059 CYWJ05 11535816 Ki = 440 nM T36059 C8P2YI 11536894 Ki = 1140 nM T36059 C0Z9UA 11536947 Ki = 699 nM T36059 CU38FS 11537425 Ki > 1000 nM T36059 CH43JG 11538373 Ki = 21 nM T36059 C5KDX9 11539152 Ki = 1030 nM T36059 CRNL17 11543615 Ki = 820 nM T36059 C1E8QF 11543839 Ki = 308 nM T36059 C16FKE 11544506 Ki > 1000 nM T36059 CW62MV 11545273 Ki = 0.44 nM T36059 CUD5B0 11546358 Ki = 110 nM T36059 CPV7Y8 11553016 Ki = 4690 nM T36059 C3IET8 11553509 Ki = 912.01 nM T36059 CHQ6F9 11554879 Ki = 8.65 nM T36059 C6CVK7 11555032 Ki = 27 nM T36059 CR70QA 11556493 Ki = 433 nM T36059 C7A9PY 11557440 Ki > 1000 nM T36059 CWR85X 11558128 Ki = 25 nM T36059 C0VES1 11560202 Ki = 10 nM T36059 CIQK94 11560605 Ki = 2.9 nM T36059 CEZJ04 11560938 Ki = 22 nM T36059 C41AXZ 11565780 Ki = 264 nM T36059 CIR70L 11565927 Ki > 1000 nM T36059 CV9N6K 11567017 Ki > 10000 nM T36059 CEH5V1 11568060 Ki >= 1000 nM T36059 C9WVP1 11568203 Ki = 408 nM T36059 C85MGW 11568359 Ki = 1083 nM T36059 CLV6H3 11568586 Ki = 2.18 nM T36059 C37CAT 11569026 Ki = 6 nM T36059 CB9TA3 11569599 Ki = 1243 nM T36059 CQB1A3 11569849 Ki = 2.58 nM T36059 CAKX79 11570379 Ki = 200 nM T36059 C54QHO 11574428 Ki >= 10000 nM T36059 C9VP0G 11574573 EC50 = 105 nM T36059 CVQ19R 11577804 Ki = 0.89 nM T36059 C5JOW8 11580374 Ki = 2370 nM T36059 CFE5O9 11584486 EC50 = 180 nM T36059 CTG7A1 11585567 Ki = 308 nM T36059 CM62BJ 11587409 Ki = 846 nM T36059 CYJ29E 11587927 Ki = 514 nM T36059 CN7T8C 11589094 Ki = 2.82 nM T36059 CL2JO8 11590539 Ki = 17.4 nM T36059 CS1RK4 11595040 Ki = 4310 nM T36059 C1ERP7 11595710 Ki = 5.5 nM T36059 C31YOR 11596733 Ki = 0.5 nM T36059 CVN1Y5 11601342 Ki > 1000 nM T36059 C1QJ4W 11602451 Ki = 2360 nM T36059 C9L7IB 11602711 Ki = 35.7 nM T36059 C80ZIV 11602914 Ki = 410 nM T36059 CAMC08 11605801 Ki = 3500 nM T36059 CLU50J 11605833 Ki = 7670 nM T36059 CAC54T 11606834 Ki = 18.2 nM T36059 CB06AO 11608818 Ki = 4640 nM T36059 C8LA0I 11609235 Ki = 3000 nM T36059 CQVZ50 11611369 Ki = 3870 nM T36059 CA5B6V 11611370 Ki = 1.63 nM T36059 C42QLP 11611903 IC50 = 0.16 nM T36059 CF09KT 11619671 Ki = 0.748 nM T36059 C31ZDE 11620703 Ki = 4020 nM T36059 C8ZIB9 11621780 Ki = 878 nM T36059 CGF25Y 11621798 Ki = 1440 nM T36059 CLV26W 11623708 Ki = 354 nM T36059 C7AM8B 11623934 Ki = 749 nM T36059 CVL8P5 11625174 Ki = 2.24 nM T36059 CJDZ72 11625255 Ki = 243 nM T36059 C2OD7U 11625772 Ki = 4.27 nM T36059 C35XDW 11625796 Ki = 12 nM T36059 CNW41M 11626796 Ki = 632 nM T36059 CA3X0M 11626875 Ki = 85.6 nM T36059 CQ2LY3 11627221 Ki = 5.2 nM T36059 C02QTY 11630237 Ki = 146.5 nM T36059 C0JOM4 11630922 Ki = 7950 nM T36059 C15AMH 11633578 Ki = 4440 nM T36059 C7TFE5 11634270 Ki = 27.8 nM T36059 CFTH84 11638790 Ki > 1000 nM T36059 C42QLC 11639150 Ki = 1610 nM T36059 CXUQ86 11640487 Ki = 2.83 nM T36059 CX4V0L 11640619 Ki > 1000 nM T36059 CM39TC 11641365 Ki = 0.81 nM T36059 C85ZEB 11642035 Ki = 10715.19 nM T36059 C37TIS 11642998 Ki = 510 nM T36059 C3VZF7 11649145 Ki = 12302.69 nM T36059 CND50M 11649544 Ki = 199 nM T36059 CT6CW3 11650023 Ki = 2.96 nM T36059 CORC41 11650245 Ki = 41.9 nM T36059 CAX46N 11654460 Ki = 56 nM T36059 C0HR7Q 11655441 Ki = 217 nM T36059 CM54YT 11657274 Ki = 3.64 nM T36059 CWY7T6 11659363 Ki = 6260 nM T36059 C1JU7A 11659696 Ki > 1000 nM T36059 C1XYR3 11659733 Ki = 82 nM T36059 CPV35M 11660022 Ki = 48 nM T36059 C4ZB9Y 11661440 Ki > 10000 nM T36059 CU94XB 11662646 Ki = 2.5 nM T36059 CV39AR 11662965 EC50 = 776 nM T36059 CQ13SY 11663152 Ki = 29.7 nM T36059 CGA72F 11663932 Ki = 0.8 nM T36059 CI2SK9 11667107 Ki > 1000 nM T36059 CGI6Y3 11667703 Ki = 11 nM T36059 CSX6B9 11674151 Ki = 51.6 nM T36059 CZ6V5H 11675684 Ki = 0.67 nM T36059 CU90TV 11675940 Ki = 5.56 nM T36059 C16PMS 11678491 Ki = 29 nM T36059 C1I6FC 11680901 Ki = 11000 nM T36059 CKU6E7 11681092 Ki = 510 nM T36059 CFD86C 11681113 Ki = 1660 nM T36059 CF54VW 11681354 Ki = 2810 nM T36059 CE8WD5 11681429 Ki = 1210 nM T36059 CI8AX3 11683024 Ki = 0.55 nM T36059 CH30ES 11684672 Ki = 9 nM T36059 CEU52V 11684979 Ki = 1.3 nM T36059 C4SWY5 11687423 Ki > 1000 nM T36059 CYFJ70 11687483 Ki = 9280 nM T36059 CI10PQ 11690712 Ki > 1000 nM T36059 CH6Q2D 11698898 Ki > 8300 nM T36059 C2V3PS 11699353 EC50 = 2520 nM T36059 CWA0C8 11701717 Ki = 135 nM T36059 CZ9IX2 11703893 Ki = 10 nM T36059 CZE9V5 11705261 Ki = 480 nM T36059 CLO6P5 11706243 Ki = 14.9 nM T36059 CR6A2V 11709311 Ki = 480 nM T36059 CX6E5A 11709650 Ki = 720 nM T36059 C8KDJ9 11710918 Ki >= 10000 nM T36059 CYI8O4 11711438 Ki = 2 nM T36059 CY48OK 11715751 Ki > 1000 nM T36059 CUM0C9 11716303 Ki = 238 nM T36059 CNR71Y 11717537 Ki = 16 nM T36059 CD72OJ 11717832 Ki = 144 nM T36059 CN6I8W 11720364 Ki = 2700 nM T36059 CH5DB1 11720501 Ki = 28 nM T36059 C4B6SX 11721301 Ki = 49200 nM T36059 C5P4YO 11723628 Ki = 4.75 nM T36059 C3ZA9B 11728558 Ki = 14.5 nM T36059 C9J4WY 11728711 Ki > 10000 nM T36059 CAMT16 11728808 Ki = 0.1799 nM T36059 CNT64M 11729275 Ki = 35 nM T36059 CR80CF 11731871 Ki > 1000 nM T36059 C5GO4E 11732736 Ki = 0.21 nM T36059 CHW0A6 11733496 Ki = 121 nM T36059 CG7Y4O 11733556 Ki = 0.4498 nM T36059 CF9Q7M 11733601 Ki = 0.7194 nM T36059 CP2J9D 11738790 Ki = 42 nM T36059 C43GFZ 11739282 Ki = 1740 nM T36059 C7OWV2 11740457 Ki = 90 nM T36059 CEVK91 11742718 Ki = 0.468 nM T36059 CYA6G4 11743031 Ki = 816 nM T36059 C0WNR6 11747281 Ki = 3020 nM T36059 CB30WZ 11756182 Ki = 8.78 nM T36059 CCU3E4 11759055 Ki = 410 nM T36059 CSR32T 11761221 Ki = 0.15 nM T36059 C7MD4U 11761823 Ki > 10000 nM T36059 CGSN15 11762418 Ki = 40 nM T36059 CI82XE 11762982 Ki = 120 nM T36059 CE1ID3 11772535 Ki = 47 nM T36059 CT84IV 11774108 Ki = 555 nM T36059 C92KBG 11776764 Ki = 2580 nM T36059 CAJ92C 11782457 Ki = 15.1 nM T36059 CO76RZ 11782906 Ki = 0.4 nM T36059 CLPT97 11784369 Ki = 1.009 nM T36059 C1TH4Z 11785771 Ki = 3510 nM T36059 C5AC6T 11792534 Ki = 12 nM T36059 C1BV0O 11794224 Ki = 201 nM T36059 CLY7D0 11795861 Ki = 8650 nM T36059 CBZJ16 11798195 Ki = 30 nM T36059 CV7T3H 11798368 Ki = 40 nM T36059 C27TPA 11798724 Ki = 296 nM T36059 CZX5B6 11799044 Ki = 229 nM T36059 CHW38G 11799536 Ki = 517 nM T36059 CL46QF 11799702 Ki = 695 nM T36059 C8ZRL4 11801496 Ki = 1258.93 nM T36059 CYN01G 11808994 Ki = 4.8 nM T36059 C3F0VS 11809235 Ki = 28.3 nM T36059 C1ZQF6 11811544 Ki = 0.7998 nM T36059 CCBY84 11811574 Ki = 75.4 nM T36059 C84NGT 11811662 Ki = 86 nM T36059 CPMB38 11811761 Ki = 1.11 nM T36059 CYE25L 11812423 Ki = 546 nM T36059 C82LEP 11812897 Ki = 3.7 nM T36059 C6ANG8 11813241 Ki > 10000 nM T36059 CZ52VY 11813713 Ki = 0.38 nM T36059 CR46ZY 11821574 Ki = 231 nM T36059 C9KMP8 11822168 Ki = 8650 nM T36059 C20MGI 11823876 Ki = 202 nM T36059 C4W2ID 11824950 Ki > 1000 nM T36059 CXBC30 11826007 Ki = 257 nM T36059 C31FGJ 11826577 Ki = 0.97 nM T36059 C15NOJ 11826924 Ki = 300 nM T36059 CT3ZH4 11834222 Ki = 2100 nM T36059 C1CQ0O 11858470 EC50 > 100000 nM T36059 CXLW54 11948707 Ki > 10000 nM T36059 CM0SL3 11956193 Ki = 660 nM T36059 C6N0YI 11957503 EC50 = 363 nM T36059 CIX09M 11962166 EC50 = 8.1 nM T36059 C0KXU5 11977965 Ki = 19 nM T36059 CXT4S5 11977966 Ki = 4120 nM T36059 CWF2B7 11977967 Ki = 380 nM T36059 CULI10 11978309 Ki = 158 nM T36059 C6Z3SF 11978310 Ki = 30 nM T36059 C1EAC3 11978313 Ki = 1420 nM T36059 CUVN07 11978421 Ki = 105 nM T36059 CE53IF 11995448 Ki > 10000 nM T36059 CUM6T1 11995557 Ki = 6700 nM T36059 CPF9I3 12066874 Ki > 10000 nM T36059 CC8Q7D 12766586 Ki = 5090 nM T36059 CW72BT 12866354 Ki = 6640 nM T36059 CM28RZ 13329020 Ki = 240 nM T36059 CWOQ92 13360944 Ki = 17000 nM T36059 CWRA96 13382931 Ki = 230 nM T36059 C1ILK4 13382932 Ki = 470000 nM T36059 CZ21VO 13382933 Ki = 86000000 nM T36059 CDF60N 13382934 Ki = 4000000 nM T36059 C5MP6U 13384165 Ki = 5100000 nM T36059 CB4M0C 13506474 Ki = 1.3 nM T36059 C24VJF 13608091 Ki = 0.91 nM T36059 C97BVY 13830108 Ki = 3.3 nM T36059 CW45MY 14040412 Ki = 13000000 nM T36059 CW7KT4 14040415 Ki = 200 nM T36059 C2K8HZ 14040416 Ki = 210000 nM T36059 CE5RM7 14040417 Ki = 240 nM T36059 CNM78X 14040418 Ki = 150 nM T36059 CV35MY 14040419 Ki = 360 nM T36059 CEAG60 14040420 Ki = 430000 nM T36059 CN13HF 14040421 Ki = 2600000 nM T36059 CCF7X0 14040422 Ki = 69 nM T36059 C6LX7C 14040423 Ki = 320000 nM T36059 CM4V6K 14086197 Ki = 64 nM T36059 CD8K6T 14157150 Ki = 569 nM T36059 CVS4J0 14426726 Ki = 376 nM T36059 CENP32 14484978 Ki = 227 nM T36059 CQS35H 14842888 Ki = 352 nM T36059 C76FZJ 14873275 Ki = 130 nM T36059 CT0IY1 14948735 Ki > 1000 nM T36059 CHO54J 14978313 Ki = 10900 nM T36059 C15GDZ 15482559 Ki = 88900 nM T36059 C9JM2H 15571954 Ki = 120 nM T36059 C65SCN 15599151 Ki = 355 nM T36059 CG0I8D 15667089 Ki = 1722 nM T36059 C8OZ5G 15667105 Ki = 2300 nM T36059 CE13QR 15729970 Ki = 370 nM T36059 CFD31U 15729977 Ki = 568 nM T36059 C5GRK6 15729982 Ki = 7270 nM T36059 CVM4T1 15926748 Ki = 326 nM T36059 C2L4NO 16037920 IC50 = 12260 nM T36059 CWFS63 16071777 Ki = 370 nM T36059 C9K2PE 16071901 Ki = 326 nM T36059 CN7F9X 16072019 Ki = 1563 nM T36059 CGX62B 16072020 Ki = 373 nM T36059 CL4ON2 16072021 Ki = 398 nM T36059 CU42YH 16072022 Ki = 4405 nM T36059 CXS8C0 16072023 Ki = 1920 nM T36059 C8W5EP 16087946 Ki = 4.3 nM T36059 CK29IS 16094546 Ki = 10.4 nM T36059 C8B5YT 16094547 Ki = 11.7 nM T36059 CM94FD 16094548 Ki = 117 nM T36059 C7FSA9 16094549 Ki = 10.3 nM T36059 C9W2FV 16094550 Ki = 9.5 nM T36059 C32PKU 16094551 Ki = 21.3 nM T36059 CF23NY 16094554 Ki = 53.9 nM T36059 CTB39W 16094555 Ki = 81.1 nM T36059 C8ZT6A 16094558 Ki = 5.6 nM T36059 C2VJ1H 16094559 Ki = 2.8 nM T36059 CA9QY7 16094561 Ki = 18 nM T36059 C18FPZ 16094562 Ki = 13.8 nM T36059 C6BI2H 16094563 Ki = 45 nM T36059 C50BPJ 16094564 Ki = 14.9 nM T36059 CQ04HA 16094565 Ki = 25.2 nM T36059 CBU5P4 16094566 Ki = 1.3 nM T36059 C3IX9U 16094567 Ki = 86.1 nM T36059 C9MO8F 16094568 Ki = 2.1 nM T36059 C7PJ9U 16094569 Ki = 1.8 nM T36059 C8X6FC 16094570 Ki = 11.5 nM T36059 C1E6YK 16094574 Ki = 11.4 nM T36059 C7DV1Q 16094575 Ki = 1.4 nM T36059 C1T7DI 16103162 Ki > 5000 nM T36059 C87PRE 16103163 Ki > 5000 nM T36059 C34YIZ 16103164 Ki > 5000 nM T36059 C6U0TL 16103165 Ki > 5000 nM T36059 CT9O5K 16103166 Ki > 5000 nM T36059 CA2W9G 16103167 Ki > 5000 nM T36059 CG74XQ 16103168 Ki > 5000 nM T36059 CL87PX 16103169 Ki = 25 nM T36059 C01PWF 16103170 Ki > 5000 nM T36059 CO3HF4 16103171 Ki > 5000 nM T36059 CIAE42 16103176 Ki > 5000 nM T36059 C0Z4KU 16103177 Ki > 5000 nM T36059 C3Y8IU 16103178 Ki > 5000 nM T36059 CA1EH0 16103179 Ki > 5000 nM T36059 CJ8O9B 16103184 Ki > 5000 nM T36059 CY3R6K 16103185 Ki > 5000 nM T36059 C9F7SM 16103186 Ki > 5000 nM T36059 C7HM0K 16103187 Ki > 5000 nM T36059 CGP93C 16115479 Ki = 5.2 nM T36059 CX4O9C 16115613 Ki = 2.8 nM T36059 CCZ67Y 16115614 Ki = 1.096 nM T36059 C4TDQ5 16115615 Ki = 3.3 nM T36059 C4EW6I 16115616 Ki = 1.9 nM T36059 C4FI6K 16115617 Ki = 3.5 nM T36059 CYKC87 16115749 Ki = 6.8 nM T36059 C4A8SU 16115750 Ki = 3.2 nM T36059 C8VXL9 16115751 Ki = 7.4 nM T36059 CRH54T 16115902 Ki = 1.7 nM T36059 C53DBK 16115903 Ki = 1.9 nM T36059 CT5UQ7 16115904 Ki = 55 nM T36059 CRZ0V4 16115905 Ki = 2.5 nM T36059 CK87MV 16115906 Ki = 1.6 nM T36059 C3G6FA 16115907 Ki = 68 nM T36059 CC53PW 16116048 Ki = 4 nM T36059 C0S1VK 16122818 Ki > 10000 nM T36059 C3KXQ7 16202724 Ki = 622 nM T36059 CFST91 16202843 Ki = 457 nM T36059 C7C3ZJ 16203430 Ki = 1340 nM T36059 C67LUN 16203541 Ki = 8730 nM T36059 CO8WS3 16203544 Ki = 599 nM T36059 CH91QO 16203667 Ki = 90 nM T36059 CTL0F3 16203668 Ki = 30 nM T36059 C4OS0D 16203669 Ki = 110 nM T36059 C0KL4A 16220189 Ki = 4.16 nM T36059 CZT4J2 16433205 Ki = 13700 nM T36059 CFE82W 16656768 Ki = 15.5 nM T36059 CSXO69 16680454 Ki = 967 nM T36059 C7WF2V 16720104 Ki > 1000 nM T36059 CT7UO9 16720105 Ki > 1000 nM T36059 C9JSW0 16720106 Ki > 1000 nM T36059 C2EPT5 16735278 Ki = 7.4 nM T36059 C5TIH3 16735279 Ki = 6.1 nM T36059 C6RT7K 16735280 Ki = 25.8 nM T36059 CVE58L 16735504 Ki = 1.66 nM T36059 C4VQ5U 16735505 Ki = 12.7 nM T36059 CNZ0D5 16735506 Ki = 24.8 nM T36059 C3XJA8 16735539 Ki = 19.9 nM T36059 C4T9HB 16735540 Ki = 3.69 nM T36059 CDV52Y 16739249 Ki = 13.9 nM T36059 C3W8DT 16749353 IC50 > 5000 nM T36059 C6AR3Q 16757019 Ki = 1180 nM T36059 CBR05N 17198004 Ki = 2 nM T36059 C2GR5M 17408222 Ki = 1000 nM T36059 CP0T2V 17427517 Ki = 1000 nM T36059 CWD1N7 17429448 Ki = 100 nM T36059 C3RTQ6 17448744 Ki = 40 nM T36059 CTA05E 17487156 Ki = 8300 nM T36059 CUW24Z 17500622 Ki = 200 nM T36059 CXH6D7 17863130 IC50 = 33 nM T36059 C8BU2E 17863131 IC50 = 320 nM T36059 CN7D2S 17863136 IC50 = 34 nM T36059 C41OLX 17863145 IC50 = 120 nM T36059 C72CYF 17863152 IC50 = 160 nM T36059 CXRL32 17863158 IC50 = 28 nM T36059 CEM6V1 17863168 IC50 = 110 nM T36059 C83NVA 17863179 IC50 = 1000 nM T36059 CIJ08G 17863186 IC50 = 140 nM T36059 CL9AX4 17863209 IC50 = 48 nM T36059 CELB65 17863210 IC50 = 260 nM T36059 C6ARU8 17863215 IC50 = 28 nM T36059 CRH9U4 17863224 IC50 = 490 nM T36059 COX01L 17863234 IC50 = 34 nM T36059 CC5YA1 18506750 Ki = 1.3 nM T36059 CBXA48 20592013 Ki = 34600 nM T36059 C5KR4S 20847387 Ki > 100000 nM T36059 C1N7ZG 20974732 Ki = 3100 nM T36059 CW50HY 20974734 Ki = 200 nM T36059 C75CPM 21128750 Ki = 211 nM T36059 CB2V8H 21603068 Ki > 100000 nM T36059 C25WAJ 21874520 Ki = 2467 nM T36059 CTK29C 21874538 Ki = 3013 nM T36059 C96PRF 21874571 Ki = 685 nM T36059 C07MZN 21874581 Ki = 340 nM T36059 C5QJC8 21874602 Ki = 530 nM T36059 CXG16I 21874603 Ki = 619 nM T36059 CV2C4F 21874613 Ki = 251 nM T36059 CB7S8A 21874626 Ki = 2576 nM T36059 CKG68C 21874634 Ki = 2224 nM T36059 CTX5P2 21874639 Ki = 2806 nM T36059 C1CKS9 21874641 Ki = 1359 nM T36059 CU80AG 21874647 Ki = 260 nM T36059 C38CXY 21874661 Ki = 1071 nM T36059 C4S5PJ 21874662 Ki = 2433 nM T36059 C14FGO 21874668 Ki = 240 nM T36059 C3WLM0 21874675 Ki = 606 nM T36059 COLC85 21874676 Ki = 1181 nM T36059 C2PZN3 21874681 Ki = 636 nM T36059 CP84GK 21874685 Ki = 285 nM T36059 CSV0W4 21874686 Ki = 752 nM T36059 CW47EF 21874687 Ki = 1019 nM T36059 C3EK0T 21874692 Ki = 1233 nM T36059 C3KH4A 21874697 Ki = 203 nM T36059 CDV73C 21874721 Ki = 450 nM T36059 C7GWD4 21874722 Ki > 10000 nM T36059 C4L8UK 21874755 Ki = 3809 nM T36059 CLY0E3 21874756 Ki = 221 nM T36059 CWQ47T 21874764 Ki = 2380 nM T36059 C74HIZ 21874771 Ki = 1138 nM T36059 C7NT1D 21874782 Ki = 123 nM T36059 CG9Y7N 21874786 Ki = 341 nM T36059 C7YRN0 21893339 Ki = 742 nM T36059 CK4HL6 21916357 Ki = 324 nM T36059 CS19AF 21916389 Ki = 35 nM T36059 CBY0E6 21916394 Ki = 326 nM T36059 CI1CO9 21916398 Ki = 107 nM T36059 CZ59CO 21916406 Ki = 160 nM T36059 C2XR0J 21916408 Ki = 204 nM T36059 C03FGL 21916419 Ki = 91 nM T36059 C4I2HN 21958524 Ki = 180 nM T36059 CKQ1C3 21958525 Ki > 9000 nM T36059 CZN1L8 21958583 Ki = 95 nM T36059 CW5NK7 21958593 Ki = 160 nM T36059 C36FJO 21958619 Ki = 262 nM T36059 CTSU04 21958681 Ki = 1500 nM T36059 CW5DG9 21958701 Ki = 1200 nM T36059 CJO62E 21958725 Ki = 110 nM T36059 C6F8TR 21958745 Ki > 9000 nM T36059 CMF03Z 21958758 Ki = 8700 nM T36059 C58MPT 21958761 Ki = 1600 nM T36059 CU7EZ3 21958783 Ki = 1100 nM T36059 CUNF42 21958814 Ki > 8300 nM T36059 C1M3OW 21989784 Ki = 2.7 nM T36059 C5HFL6 22002319 Ki = 282 nM T36059 CFH75K 22002352 Ki = 159 nM T36059 C02SLQ 22002364 Ki = 38.7 nM T36059 CPS61Y 22002375 Ki = 609 nM T36059 C3CV9X 22002449 Ki = 238 nM T36059 CKME84 22055296 Ki = 9 nM T36059 C43TSO 22055299 Ki = 25 nM T36059 C7CW3I 22266730 Ki = 2117 nM T36059 CZF4S2 22266732 Ki > 9000 nM T36059 CTO91Z 22266738 Ki = 3300 nM T36059 CC2N6M 22266741 Ki > 9000 nM T36059 CZL43T 22266742 Ki > 9000 nM T36059 CV6E4A 22266746 Ki = 92 nM T36059 CU16OK 22266751 Ki > 9000 nM T36059 C2QUH0 22266756 Ki > 9000 nM T36059 CIOB39 22266761 Ki > 9000 nM T36059 CC12SJ 22266763 Ki = 2300 nM T36059 C4ZJ1F 22266765 Ki = 630 nM T36059 C3WK8Z 22266766 Ki > 9000 nM T36059 CAGC71 22266769 Ki = 3810 nM T36059 CV53YM 22266771 Ki > 9000 nM T36059 CSC37U 22266775 Ki = 1800 nM T36059 CCQ0I1 22266776 Ki > 9000 nM T36059 CDWI49 22266778 Ki = 453 nM T36059 CC94DE 22266784 Ki = 1800 nM T36059 C7G0LF 22282339 Ki = 0.36 nM T36059 CJ52EV 23371936 Ki = 6140 nM T36059 CW1M6N 23523299 Ki = 130 nM T36059 CF5S9T 23643558 EC50 = 11.2 nM T36059 C3XM6N 23643659 EC50 = 3.8 nM T36059 C8IU6O 23653582 IC50 = 8.2 nM T36059 C65SJK 23656931 Ki = 368.5 nM T36059 CGRT64 23656932 Ki = 29.2 nM T36059 C8N0LF 23656933 Ki = 557.3 nM T36059 CYU94Z 23656934 Ki = 101.2 nM T36059 C8SC3A 23656935 Ki = 15 nM T36059 CO98NZ 23656936 IC50 = 0.58 nM T36059 CV28WL 23656937 Ki > 1000 nM T36059 CAG3Y8 23657103 Ki = 9.2 nM T36059 CKRG98 23657104 Ki = 49.1 nM T36059 C6YS2Z 23657105 Ki = 34.6 nM T36059 CZ6H4G 23657106 Ki = 33.2 nM T36059 C6F4UV 23657107 Ki = 51 nM T36059 C26AWG 23657108 Ki = 295.2 nM T36059 C0R9DW 23657109 Ki = 103 nM T36059 COD51S 23657262 Ki = 4.3 nM T36059 CSZB58 23657263 Ki = 55.7 nM T36059 C68QBD 23657264 Ki = 41.5 nM T36059 C1SWM6 23657265 Ki = 1.6 nM T36059 CG4I1H 23657266 IC50 = 11.61 nM T36059 CMSG38 23657267 Ki = 97 nM T36059 C6GDP9 23657408 Ki = 49 nM T36059 CVBI12 23657409 Ki = 43.4 nM T36059 CRY24K 23702720 Ki = 183 nM T36059 CFE2N1 23757284 Ki = 0.75 nM T36059 CVO53U 23900137 Ki = 5.5 nM T36059 CM2KN8 24749593 Ki = 87.5 nM T36059 CJ3QZ4 24749594 Ki = 98.3 nM T36059 C8A4PO 24749597 Ki = 19.5 nM T36059 C7Q9LM 24749599 Ki = 26.7 nM T36059 C2X9TI 24749600 Ki = 27.2 nM T36059 CEA0J5 24768437 Ki = 31 nM T36059 C8NKT5 24768438 Ki = 45 nM T36059 C5FJU3 24768439 Ki = 166 nM T36059 CS85OX 24768440 Ki = 276 nM T36059 C2U5TQ 24768441 Ki = 26 nM T36059 CGVO15 24768442 Ki = 38 nM T36059 C3GM4B 24768443 Ki = 525 nM T36059 CSJW71 24768444 Ki = 7.5 nM T36059 C53BPO 24768445 Ki = 6.3 nM T36059 CYZI26 24768446 Ki = 7.1 nM T36059 CD1C5T 24768447 Ki = 3.5 nM T36059 CX7W5M 24768448 Ki = 30 nM T36059 C90QOD 24768449 Ki = 1.8 nM T36059 C06UBG 24768450 IC50 = 1.25 nM T36059 CR32ME 24768451 Ki = 22 nM T36059 C09WQS 24768452 IC50 = 1.84 nM T36059 C6S1HG 24810000 Ki > 557 nM T36059 CK02ZF 24812771 Ki = 19 nM T36059 CK8J3I 24824328 Ki = 8.6 nM T36059 CKC0W3 24827442 Ki = 250 nM T36059 CIR6E9 24827552 Ki = 290 nM T36059 C15VIG 24827553 Ki = 440 nM T36059 C06PBV 24827554 Ki = 350 nM T36059 C34RNS 24827555 Ki = 400 nM T36059 CWPS95 24828457 Ki = 950 nM T36059 CU0Q2I 24878975 Ki = 0.92 nM T36059 C05BYL 24882472 Ki > 100000 nM T36059 CU24RD 24950533 Ki = 390 nM T36059 C0YGQ2 24998410 Ki = 526 nM T36059 C2EK5G 25002987 Ki = 7.3 nM T36059 COSA97 25003338 Ki = 1.5 nM T36059 C7DF0O 25003339 Ki = 6.8 nM T36059 C1ZXW0 25003340 Ki = 1.5 nM T36059 CHEX21 25003341 Ki = 13 nM T36059 CL5NI4 25008276 Ki = 9.32 nM T36059 CW5YA6 25066016 Ki = 945 nM T36059 CK92QL 25070230 Ki = 63.1 nM T36059 CAX68Y 25104834 Ki = 92 nM T36059 CP5RY7 25104946 Ki = 5608 nM T36059 CX63TW 25129539 Ki = 4.8 nM T36059 C7JE1V 25147618 Ki = 38 nM T36059 C5FHU3 25147619 Ki = 34 nM T36059 CN2FL7 25188209 Ki = 2108 nM T36059 C9V4RO 25212375 Ki = 3.4 nM T36059 CA28TU 25212376 Ki = 5 nM T36059 CFR20P 25223817 Ki = 2.5 nM T36059 CY18BR 25573285 Ki = 3000 nM T36059 C29JQB 25617525 Ki = 5300 nM T36059 CS0V9B 32178888 Ki = 2600 nM T36059 C8DT0B 32459044 Ki = 1900 nM T36059 CJ95TD 32459103 Ki = 2200 nM T36059 CFW2X3 32459568 Ki = 1400 nM T36059 CSE07H 32459683 Ki = 5500 nM T36059 C4MB8S 32460014 Ki = 1900 nM T36059 C3FH2I 32460336 Ki = 2600 nM T36059 C6LI7R 32460717 Ki = 600 nM T36059 C7Z2BV 32460731 Ki = 300 nM T36059 C01BKR 32460889 Ki = 2300 nM T36059 C6VG3H 32461058 Ki = 500 nM T36059 CU51PG 32461094 Ki = 1500 nM T36059 C4OUE0 32461100 Ki = 2700 nM T36059 C8TE4D 32461405 Ki = 3300 nM T36059 CKS89N 32461556 Ki = 2500 nM T36059 CWUA82 42625614 Ki = 6740 nM T36059 C6W4XM 42625615 Ki = 3030 nM T36059 CX8DV9 42625691 Ki = 1440 nM T36059 C5I8NE 42625766 Ki = 479 nM T36059 CIG29P 42625767 Ki = 1150 nM T36059 C4SL9A 42625923 Ki = 251 nM T36059 C4NS7C 42625924 Ki = 3.3 nM T36059 C9FLC8 42626000 Ki = 158 nM T36059 CETQ95 42626002 Ki = 15.5 nM T36059 CBW7G5 42626003 Ki = 8.4 nM T36059 C6RIC7 42626004 Ki = 70.3 nM T36059 C4Y7NP 42626075 Ki = 41 nM T36059 CE2QT0 42626076 Ki = 335 nM T36059 C1LC2U 42626077 Ki = 7.75 nM T36059 C7OSK6 42626153 Ki = 590 nM T36059 C2X5MR 42626155 Ki = 656 nM T36059 C3UQR6 42626156 Ki = 490 nM T36059 C16MHP 42626157 Ki = 1335 nM T36059 C8FG0O 42626158 Ki = 138 nM T36059 C8RDW2 42626220 Ki = 11.7 nM T36059 CLE2K9 42626221 Ki = 4.54 nM T36059 CTBW80 42636897 Ki = 1290 nM T36059 C1J6SG 44185870 Ki = 434 nM T36059 C3OXF9 44185872 Ki > 1000 nM T36059 CS9Q4K 44185873 Ki > 1000 nM T36059 CX24EI 44185874 Ki > 1000 nM T36059 CWH1S5 44185932 Ki > 1000 nM T36059 CWX1B7 44185933 Ki > 1000 nM T36059 CF2K1H 44185934 Ki = 209 nM T36059 C8PMD7 44185935 Ki = 140 nM T36059 C8I9LD 44185936 Ki = 2080 nM T36059 CQRH91 44186579 Ki > 10000 nM T36059 C9RG0P 44186580 Ki > 10000 nM T36059 C48XKD 44186582 Ki = 557 nM T36059 CCNH98 44186622 Ki = 24200 nM T36059 CY2D4F 44186623 Ki > 1000 nM T36059 CRWD47 44186624 Ki = 758 nM T36059 CAY95F 44186625 Ki = 5780 nM T36059 C42DUI 44186626 Ki > 1000 nM T36059 CYE0X8 44186667 Ki > 10000 nM T36059 CM7B3X 44186668 Ki > 10000 nM T36059 C69VCO 44186669 Ki = 30000 nM T36059 CSBP65 44186670 Ki > 1000 nM T36059 CZJ29Y 44186715 Ki = 156 nM T36059 C5X9NC 44186716 Ki > 1000 nM T36059 C6JG3Q 44186717 Ki > 10000 nM T36059 CE21OP 44186718 Ki > 10000 nM T36059 C9W0OQ 44186719 Ki = 17600 nM T36059 C59XNK 44203236 Ki = 131 nM T36059 CIL82A 44203643 Ki = 18.3 nM T36059 CWS89X 44203645 Ki = 25.3 nM T36059 C84FSP 44203646 Ki = 1903 nM T36059 C2NDY3 44203648 Ki = 11 nM T36059 CC35JG 44219683 Ki = 1288.25 nM T36059 CXIT13 44219684 Ki = 398.11 nM T36059 C0SBK7 44232535 Ki = 2.38 nM T36059 CK1H5B 44241696 Ki = 3.82 nM T36059 C7Z4RE 44275982 Ki = 84.7 nM T36059 CSW1E4 44275995 Ki = 29.9 nM T36059 CD2I6F 44276002 Ki = 2880 nM T36059 CP5M2R 44276273 Ki = 1090 nM T36059 C8TJ7M 44276306 Ki = 912 nM T36059 CU35RG 44276349 Ki = 22.5 nM T36059 C7T0ZY 44281663 Ki > 1000 nM T36059 CX3YV9 44281684 Ki > 1000 nM T36059 CJ3QM8 44281700 Ki > 1000 nM T36059 CN72HK 44281738 Ki > 1000 nM T36059 C7HV4D 44284007 Ki = 1010 nM T36059 CL8XS1 44284052 Ki = 1060 nM T36059 C28QCM 44284065 Ki = 2760 nM T36059 C8YHM6 44284095 Ki = 2710 nM T36059 CUR2Q6 44284189 Ki = 1230 nM T36059 CE5V1M 44284209 Ki = 1410 nM T36059 CBQ90F 44284222 Ki = 1040 nM T36059 C34FVI 44284223 Ki = 181 nM T36059 CT0EV8 44284345 Ki = 900 nM T36059 C7O5MJ 44309799 Ki = 1960 nM T36059 C7W3OA 44311416 Ki = 71 nM T36059 CWD4M1 44311471 Ki = 172 nM T36059 CTY68F 44313377 Ki = 1860 nM T36059 CLS37N 44313528 Ki = 19000 nM T36059 C35XPZ 44313794 Ki = 4350 nM T36059 C8ZBR6 44313808 Ki = 561 nM T36059 C1K9LU 44341299 Ki = 555 nM T36059 C1K5YL 44343643 Ki = 3330 nM T36059 C2U4CB 44343895 IC50 = 27.54 nM T36059 C8V6QA 44344926 Ki = 72 nM T36059 C4YMS3 44351802 Ki = 7800000 nM T36059 CZ39AT 44352279 Ki = 2300000 nM T36059 C0PO2B 44354130 Ki = 1.4 nM T36059 CPU06D 44359213 EC50 = 1.4 nM T36059 C0IT5W 44359214 Ki = 46 nM T36059 CSQF92 44359257 Ki = 490 nM T36059 CYG81L 44359364 Ki = 1.2 nM T36059 C3ML1G 44377565 Ki = 1200 nM T36059 C36UAM 44379939 Ki = 1 nM T36059 CX4K8P 44380438 Ki = 75 nM T36059 CO78DN 44387284 Ki = 1.5 nM T36059 CJ85QM 44388202 Ki = 21 nM T36059 CPZ64O 44388205 Ki = 163 nM T36059 CT9I2W 44388206 Ki = 15 nM T36059 CCJT49 44388207 Ki = 55 nM T36059 CHU5R2 44388211 Ki = 65 nM T36059 CC02XN 44388218 Ki = 1480 nM T36059 C84SKL 44388222 Ki = 39 nM T36059 C1T2FP 44388225 Ki = 2488 nM T36059 CP76KB 44388242 Ki = 8.995 nM T36059 C3L2EW 44388246 Ki = 4.898 nM T36059 CF9AL1 44388252 Ki = 65 nM T36059 CBZ2P1 44390545 Ki = 39 nM T36059 C83KXG 44396444 Ki = 3 nM T36059 C7K1ST 44396450 Ki = 6 nM T36059 C4AOY9 44396470 Ki = 170 nM T36059 C32JTS 44396478 Ki = 2 nM T36059 CHY08U 44396487 Ki = 320 nM T36059 CS0D8B 44396500 Ki = 157 nM T36059 C8B1XJ 44396515 Ki = 10 nM T36059 CXZ7Q4 44396516 Ki = 109 nM T36059 CY7B3D 44396545 Ki = 19 nM T36059 C7ERK1 44396546 Ki = 60 nM T36059 CH3KV6 44396553 Ki = 148 nM T36059 C8D0HQ 44396598 Ki = 49 nM T36059 C0N1FZ 44396599 Ki = 97 nM T36059 CHT68B 44397718 Ki = 1460 nM T36059 C4TU8O 44397776 Ki = 122 nM T36059 C5V8UZ 44397952 Ki = 1570 nM T36059 C4QNR0 44401051 Ki = 42 nM T36059 CXCE96 44401487 Ki = 0.86 nM T36059 C5U2YX 44401545 Ki = 4.5 nM T36059 CT7W3U 44401604 Ki = 39 nM T36059 CXHS76 44402758 Ki = 134 nM T36059 CV8BG5 44402784 Ki = 419 nM T36059 C24THP 44405058 Ki = 673 nM T36059 CTE46U 44405094 Ki = 229 nM T36059 C6K2YX 44405115 Ki = 111 nM T36059 C54JHF 44405119 Ki = 163 nM T36059 CTG2S3 44405123 Ki = 396 nM T36059 CB3X0L 44405124 Ki = 104.2 nM T36059 CN94AX 44406328 Ki = 3000 nM T36059 C3JPG9 44406334 Ki = 4900 nM T36059 C3S9CP 44406397 Ki = 4400 nM T36059 CAF1Y3 44406398 Ki = 4200 nM T36059 CT21RA 44406403 Ki > 5000 nM T36059 CA8FV4 44406545 Ki = 490 nM T36059 CG8MQ9 44406555 Ki = 410 nM T36059 CUPC05 44406556 Ki = 1500 nM T36059 C5ZW8S 44406562 Ki = 600 nM T36059 CQ98MC 44406567 Ki = 620 nM T36059 CN7V0Y 44406570 Ki = 2300 nM T36059 CI19OT 44406582 Ki = 970 nM T36059 CZPM65 44406588 Ki = 2000 nM T36059 C6O9TH 44406592 Ki = 340 nM T36059 CJA23V 44406607 Ki = 330 nM T36059 CV5AO7 44406611 Ki = 640 nM T36059 CE3CP9 44406617 Ki = 960 nM T36059 CVQ2B8 44406625 Ki = 3000 nM T36059 CD9E7F 44406639 Ki = 1300 nM T36059 CK7GF1 44406642 Ki = 950 nM T36059 CPEV01 44406643 Ki = 490 nM T36059 CK9ZB7 44407518 Ki = 315 nM T36059 CES29R 44408316 Ki = 3.5 nM T36059 C0EB9D 44410399 Ki = 3.77 nM T36059 C6E4RA 44410402 Ki = 2.03 nM T36059 C5IVA3 44410403 Ki = 1.91 nM T36059 CI7W8R 44410406 Ki = 1.31 nM T36059 CWQX21 44410409 Ki = 1.98 nM T36059 CJ26LR 44410410 Ki = 27.2 nM T36059 CG30RK 44410412 Ki = 6.05 nM T36059 CC54QX 44410479 Ki = 390 nM T36059 C04CDS 44410480 Ki > 3000 nM T36059 CSO5B3 44410523 Ki > 3000 nM T36059 CK8I1V 44410544 Ki = 1.28 nM T36059 CO2LJ0 44410545 Ki = 2.4 nM T36059 CX9OZ0 44410549 Ki = 4.58 nM T36059 C7DER1 44410550 Ki = 1.29 nM T36059 C6E8OT 44410551 Ki = 1.6 nM T36059 CZ94PN 44410554 Ki = 3.45 nM T36059 COWL13 44410555 Ki = 1.35 nM T36059 CHU6Q0 44410556 Ki = 2.22 nM T36059 CVYF89 44410559 Ki = 20.1 nM T36059 C2YF8L 44410561 Ki = 2.13 nM T36059 CXD2R9 44410566 Ki = 1.17 nM T36059 C0AU8J 44410580 Ki = 25 nM T36059 C20FJQ 44410585 Ki = 2.42 nM T36059 CZP52D 44410590 Ki = 709 nM T36059 CQ8E2B 44410597 Ki = 0.754 nM T36059 C0P5FH 44410636 Ki = 2700 nM T36059 CYG5K3 44410655 Ki = 1.02 nM T36059 CY2R8U 44410673 Ki = 1500 nM T36059 C02UCY 44410674 Ki = 20 nM T36059 C41KLQ 44410684 Ki = 6.2 nM T36059 C8DE9A 44410690 Ki = 0.709 nM T36059 CSTP07 44410691 Ki = 0.542 nM T36059 CV37TH 44410697 Ki = 1.84 nM T36059 C5M4TE 44410739 Ki = 3.9 nM T36059 CWT7J5 44410740 Ki = 59 nM T36059 C6ZML8 44410744 Ki = 87 nM T36059 C8OR7G 44410745 Ki > 3000 nM T36059 CEY8N2 44410750 Ki = 6.8 nM T36059 CSOB71 44410754 Ki = 18 nM T36059 C1RI8K 44410761 Ki = 140 nM T36059 CQ4DF8 44410819 Ki = 9.1 nM T36059 C4NY6I 44410846 Ki = 110 nM T36059 CC6SR4 44410847 Ki = 700 nM T36059 C0DXE8 44413083 Ki = 120 nM T36059 CSLZ52 44413084 Ki = 8.3 nM T36059 CV9C5B 44413096 IC50 = 18950 nM T36059 CV2KP9 44413097 Ki = 19 nM T36059 C58DGO 44413098 Ki = 7.9 nM T36059 CNDQ05 44413106 IC50 = 950 nM T36059 CN4W1C 44413108 Ki = 20 nM T36059 C7PAD9 44413113 IC50 = 21880 nM T36059 C37HYD 44413131 Ki = 380 nM T36059 C1PI5R 44413182 IC50 = 38050 nM T36059 CMT4W9 44413192 IC50 = 7600 nM T36059 C2ZH7P 44413202 IC50 = 14860 nM T36059 CT1Y7P 44413313 Ki = 260 nM T36059 CZ3XT4 44413359 Ki = 0.14 nM T36059 C9D6SN 44413380 Ki = 0.86 nM T36059 CN51SA 44413381 Ki = 0.56 nM T36059 COD4F9 44417680 Ki = 4810 nM T36059 CSR4Q2 44420921 Ki = 93.3 nM T36059 CWJ19B 44420922 Ki = 101 nM T36059 CO68UH 44420926 Ki = 5.1 nM T36059 CUE35G 44420928 Ki = 312 nM T36059 C1V0HC 44420930 Ki = 77.8 nM T36059 C01VYU 44420931 Ki = 119 nM T36059 C3C8LS 44423811 Ki = 38.4 nM T36059 CWCH32 44423812 Ki = 72.3 nM T36059 CDY6P7 44423813 Ki = 34.2 nM T36059 CYR14N 44423814 Ki = 36.4 nM T36059 C2F3DE 44423815 Ki = 85.2 nM T36059 CF26JD 44423816 Ki = 115 nM T36059 CE76XB 44423817 Ki = 25.3 nM T36059 C5J3PM 44423818 Ki = 53.2 nM T36059 CA2HW6 44423819 Ki = 78.6 nM T36059 CFM1I4 44423820 Ki = 81.4 nM T36059 CFTE30 44423821 Ki = 40.2 nM T36059 CQL6J8 44423822 Ki = 320 nM T36059 C4QFX3 44423823 Ki = 42.3 nM T36059 CWQK67 44423824 Ki = 82.7 nM T36059 CG5O9I 44423825 Ki = 65.4 nM T36059 CK1EQ6 44423826 Ki = 72.5 nM T36059 C4ZL9F 44423827 Ki = 107 nM T36059 CH96WQ 44423828 Ki = 101 nM T36059 CLJ9T4 44423837 Ki = 75.7 nM T36059 CT1YQ4 44423838 Ki = 95.8 nM T36059 C49JVO 44427579 Ki = 7.3 nM T36059 CID63L 44427580 Ki = 85.5 nM T36059 CWL9P8 44427581 Ki = 228.5 nM T36059 CG5C8V 44427582 Ki = 31 nM T36059 CVA8F6 44427583 Ki = 123 nM T36059 CGM8E6 44427584 Ki = 101.5 nM T36059 C7L2KY 44427585 Ki = 4.3 nM T36059 C3Q1BN 44427586 Ki = 4.4 nM T36059 C91TWO 44427587 Ki = 3.4 nM T36059 CX1KI5 44427588 Ki = 3.9 nM T36059 CYM3S8 44427589 Ki = 5.6 nM T36059 C6BPF4 44427590 Ki = 4.5 nM T36059 C4FLS1 44427591 Ki = 14 nM T36059 CG5PI2 44427592 Ki = 11.5 nM T36059 C6SCA9 44427594 Ki = 9 nM T36059 C1GY3X 44427595 Ki = 3.35 nM T36059 CV3O9J 44427596 Ki = 257 nM T36059 CWO87J 44427598 Ki = 6.1 nM T36059 CNB2O5 44427599 Ki = 23.25 nM T36059 CGR07Z 44427600 Ki = 30 nM T36059 C7PT2S 44430151 Ki = 107 nM T36059 CBW73G 44430154 Ki = 41 nM T36059 CDU4P8 44430156 Ki = 710 nM T36059 CA9L1D 44430158 Ki = 132 nM T36059 C9M0OF 44430160 Ki = 49 nM T36059 C0HBJ8 44430163 Ki = 3210 nM T36059 CQF30M 44430165 Ki = 54 nM T36059 C2F3ZV 44430169 Ki = 15 nM T36059 C4IT7U 44430170 Ki = 4 nM T36059 C4S5DC 44430171 Ki = 92 nM T36059 CYS8I1 44430173 Ki = 3160 nM T36059 CLW6M5 44430177 Ki = 20 nM T36059 CZ2CX5 44430187 Ki = 250 nM T36059 C42LMQ 44430188 Ki > 5000 nM T36059 C0UDY1 44430192 Ki = 1270 nM T36059 C87TZB 44430198 Ki = 94 nM T36059 CI97LW 44430203 Ki = 15 nM T36059 CPW14D 44430206 Ki = 3 nM T36059 CNX54A 44430209 Ki = 4 nM T36059 CC20AB 44430231 Ki = 26 nM T36059 C09MBQ 44430232 Ki = 36 nM T36059 CDH26R 44430235 Ki = 63 nM T36059 C8UN2W 44430236 Ki = 77 nM T36059 CX5RU6 44430239 Ki = 0.7 nM T36059 CL6C1D 44430241 Ki = 0.57 nM T36059 CHA27B 44436074 EC50 > 100000 nM T36059 C7CN4U 44436075 EC50 > 100000 nM T36059 CUXK23 44436076 IC50 = 150 nM T36059 CX57KM 44436077 EC50 > 100000 nM T36059 CQ79OA 44436078 IC50 = 170 nM T36059 C1TB8X 44436079 IC50 = 12 nM T36059 CWSJ63 44436080 EC50 = 453 nM T36059 CNX39I 44436082 EC50 = 1.9 nM T36059 CL7R5B 44437222 Ki > 1000 nM T36059 CIBX81 44437223 Ki > 1000 nM T36059 CLHJ58 44437228 Ki > 1000 nM T36059 CCS1Z4 44437229 Ki > 1000 nM T36059 CC1FS6 44437230 Ki > 1000 nM T36059 C5QIO9 44437231 Ki > 1000 nM T36059 CGWI08 44437232 Ki > 1000 nM T36059 C67ZNA 44437460 Ki = 15200 nM T36059 C92FBY 44437466 Ki > 10000 nM T36059 CD83GF 44437468 Ki = 1600 nM T36059 C34KTJ 44437470 Ki = 1290 nM T36059 CYB86Z 44442015 Ki = 280 nM T36059 C1UIO8 44442016 Ki = 25000 nM T36059 CUP5T0 44442018 Ki = 14 nM T36059 C4RDK6 44442019 Ki = 84 nM T36059 CPC63E 44442162 Ki = 790 nM T36059 C71XQS 44442163 Ki = 8560 nM T36059 C42ZRD 44442166 Ki = 89 nM T36059 C9Z3CW 44442167 Ki = 7 nM T36059 C06RLU 44446477 Ki = 1000 nM T36059 CFPZ19 44447519 Ki > 100000 nM T36059 CJ7MS5 44447534 Ki > 100000 nM T36059 C3LOJ1 44447535 Ki > 100000 nM T36059 C64RXH 44448951 Ki = 5.21 nM T36059 C6SF2I 44448952 Ki = 2.88 nM T36059 C05ZJG 44448978 Ki = 149 nM T36059 CJ4DM9 44448979 Ki = 17.1 nM T36059 C74XLS 44448982 Ki = 2.17 nM T36059 CVEX70 44449007 Ki = 1.17 nM T36059 CJ8N1Z 44449034 Ki = 0.82 nM T36059 CPL2F0 44449058 Ki = 0.98 nM T36059 CJLF50 44449113 Ki = 1.3 nM T36059 CP7Z2O 44449141 Ki = 1.3 nM T36059 CME34Q 44449532 Ki = 456 nM T36059 CZUB58 44449635 Ki = 1759 nM T36059 CHP5W0 44450290 Ki = 1.4 nM T36059 CN7TA8 44451127 Ki = 2238.72 nM T36059 CQT8F6 44451144 Ki = 60 nM T36059 CYOF07 44451499 Ki = 30.7 nM T36059 CO0UD1 44451500 Ki = 53.9 nM T36059 CGS85Y 44451501 Ki = 634 nM T36059 CL8PQ6 44451524 Ki = 186 nM T36059 C1KXG7 44452431 Ki = 251.19 nM T36059 C6AG2Y 44452434 Ki = 100 nM T36059 CJW91V 44452435 Ki = 125.89 nM T36059 C87QHW 44452454 Ki = 676.08 nM T36059 C0PER5 44452455 Ki = 251.19 nM T36059 CI5HT1 44452456 Ki = 1548.82 nM T36059 CK16BV 44452457 Ki = 66.07 nM T36059 CG74SF 44452515 Ki = 436.52 nM T36059 C18BXC 44452535 Ki = 30.2 nM T36059 CWF9E6 44452536 Ki = 22.91 nM T36059 CSFV93 44452539 Ki = 371.54 nM T36059 C4B7VM 44454763 Ki = 867 nM T36059 C2EQM1 44454764 Ki = 1530 nM T36059 CWZG75 44454788 Ki = 117 nM T36059 C9YD4Q 44454789 Ki = 43.4 nM T36059 CN7Y2F 44454816 Ki = 667 nM T36059 CTWR48 44454817 Ki = 398 nM T36059 CU5XL2 44454818 Ki = 565 nM T36059 CB67EY 44454849 Ki = 126 nM T36059 C60CIT 44454850 Ki = 837 nM T36059 CZU8C6 44454851 Ki = 727 nM T36059 CH5SW9 44454853 Ki = 115 nM T36059 CL39AN 44454883 Ki = 30.7 nM T36059 C7UK9H 44454885 Ki = 425 nM T36059 C52HBA 44454886 Ki = 109 nM T36059 C7APO0 44454922 Ki = 136 nM T36059 C52LGN 44454923 Ki = 21.3 nM T36059 C6CO9J 44454925 Ki = 121 nM T36059 C9JL7N 44457461 Ki = 3190 nM T36059 CXOS03 44457466 Ki = 332 nM T36059 C6A9OT 44457469 Ki = 526 nM T36059 CS1F5E 44457473 Ki = 13.9 nM T36059 CR58PU 44457922 Ki > 10000 nM T36059 CIDT05 44457923 Ki > 10000 nM T36059 C0GTF5 44457953 Ki > 10000 nM T36059 C2GTV4 44458220 Ki > 10000 nM T36059 CZ70PN 44461607 Ki = 557 nM T36059 C4DL5C 44469677 IC50 = 1 nM T36059 CB7K2Y 44520941 Ki = 896 nM T36059 CZ6F9S 44520976 Ki = 366 nM T36059 CQ71XC 44520980 Ki = 1150 nM T36059 CEO4P7 44520981 Ki = 9090 nM T36059 C31SUP 44520982 Ki = 2104 nM T36059 CNR53B 44520983 Ki = 741 nM T36059 C3MZC5 44520985 Ki = 1627 nM T36059 CJ57RW 44537897 Ki = 266 nM T36059 CV14GL 44562752 Ki = 50 nM T36059 CLI7K5 44562753 Ki = 7.5 nM T36059 CWJ0Q1 44562754 Ki = 50 nM T36059 CE5K2G 44562755 Ki = 40 nM T36059 CVW3N2 44563977 Ki = 1 nM T36059 CV6I0P 44567439 Ki = 43400 nM T36059 C2RJ7Q 44568838 Ki = 0.25 nM T36059 CJ7M4D 44570108 Ki = 60 nM T36059 C6LX7E 44570109 Ki = 15.5 nM T36059 C1MB5K 44570110 Ki = 10.5 nM T36059 CJG71E 44570111 Ki = 945 nM T36059 C19ZCI 44570154 Ki = 210 nM T36059 C5YTX8 44570155 Ki = 65 nM T36059 C0S5EM 44570156 Ki = 11.5 nM T36059 C5QH3R 44570157 Ki = 24.7 nM T36059 CI2ED7 44570158 Ki = 52 nM T36059 CAD27U 44570195 Ki = 140 nM T36059 C1U6VP 44570196 Ki = 60 nM T36059 CI43PN 44570197 Ki = 415 nM T36059 CG4XP9 44570198 Ki = 6.3 nM T36059 CKOC54 44570242 Ki = 11.5 nM T36059 CO2A4G 44570248 Ki = 480 nM T36059 CW0B5D 44570367 Ki = 141 nM T36059 C9BA3H 44570369 Ki = 57 nM T36059 C24CRG 44570413 Ki = 182 nM T36059 C6EAT9 44570414 Ki = 148 nM T36059 CTS6P4 44570415 Ki = 110 nM T36059 CP93SE 44570416 Ki = 5.13 nM T36059 C6NJP3 44570454 Ki = 15 nM T36059 CC6TW2 44570455 Ki = 20 nM T36059 CG9BR2 44570456 Ki = 98 nM T36059 C9FV0G 44570457 Ki > 1000 nM T36059 CC51RV 44570458 Ki > 1000 nM T36059 CSMN18 44570493 Ki = 200 nM T36059 CMD87Q 44572294 Ki > 100000 nM T36059 CSL0G8 44572353 Ki > 100000 nM T36059 C0ETQ1 44572354 Ki > 100000 nM T36059 C7D2GC 44572410 Ki > 100000 nM T36059 C9VS8P 44572470 Ki > 100000 nM T36059 CDZ14G 44572472 Ki > 100000 nM T36059 C3N5UW 44572536 Ki = 279 nM T36059 C4YE2H 44572580 Ki = 281 nM T36059 C8Y0EI 44574117 Ki = 275 nM T36059 CZDG39 44574118 Ki = 871 nM T36059 CZX7N5 44574165 Ki = 363 nM T36059 CUH78B 44574194 Ki = 331 nM T36059 CMFB42 44574222 Ki = 71 nM T36059 CA31JY 44579667 Ki = 12.4 nM T36059 CR0GX1 44579668 Ki = 86.2 nM T36059 C7RA4N 44579669 Ki = 70.2 nM T36059 C2TZQ6 44579670 Ki = 310 nM T36059 CZS2C8 44579671 Ki = 196 nM T36059 CCN45J 44579672 Ki = 1010 nM T36059 CF04WK 44579673 Ki = 1.58 nM T36059 CRS81G 44579674 Ki = 4.06 nM T36059 CF2O3K 44579675 Ki = 1.3 nM T36059 CL18FO 44579714 Ki = 1.44 nM T36059 C5TKU6 44579715 Ki = 1.06 nM T36059 CI4FW1 44579716 Ki = 0.73 nM T36059 CZ7NV2 44579717 Ki = 1.42 nM T36059 CCB34Q 44582614 Ki = 1410 nM T36059 CSM58E 44582652 Ki = 11600 nM T36059 CA5R4M 44582653 Ki = 5900 nM T36059 CR95SV 44582654 Ki = 296 nM T36059 C8G4TH 44582690 Ki = 3480 nM T36059 CV5F9X 44582691 Ki = 4350 nM T36059 C71SDJ 44582723 Ki = 746 nM T36059 CLW60K 44582724 Ki = 2520 nM T36059 CH07JS 44582725 Ki = 4490 nM T36059 CZ91EO 44582726 Ki = 129 nM T36059 C9Y8VU 44583006 Ki > 10000 nM T36059 CR3LW0 44583035 Ki > 1000 nM T36059 CS5MA2 44586053 Ki = 1370 nM T36059 CJ8P2X 44586198 Ki = 32.2 nM T36059 C7D9YB 44586199 Ki = 2.2 nM T36059 C71NOS 44586200 Ki = 100 nM T36059 C36YLB 44586201 Ki = 1427 nM T36059 CS6IH5 44586225 Ki = 493 nM T36059 CI1VJ4 44586227 Ki = 5.5 nM T36059 C9U6XI 44586228 Ki = 387 nM T36059 CY2MH0 44586253 Ki = 83.5 nM T36059 CY03KI 44586254 Ki = 65 nM T36059 C05QFY 44586255 Ki = 63 nM T36059 C9XOP5 44586256 Ki = 1300 nM T36059 C1LR0F 44586296 Ki = 953 nM T36059 C9P6WK 44586297 Ki = 21 nM T36059 CI1Y7G 44586298 Ki = 6.4 nM T36059 CC7FH5 44586717 Ki = 68 nM T36059 C7S1MY 44586718 Ki = 6.1 nM T36059 C6IO7C 44587956 Ki = 1290 nM T36059 CUG8E4 44587957 Ki = 891 nM T36059 CG1JD0 44588395 Ki = 182 nM T36059 CBL10K 44588516 Ki = 295 nM T36059 CU0B3W 44590253 Ki = 103 nM T36059 CW7UO3 44590255 Ki = 5531 nM T36059 C1UL3Z 44590290 Ki = 4852 nM T36059 C0D8HM 44590292 Ki = 4107 nM T36059 CU1Q2X 44590384 Ki = 560 nM T36059 C03OBL 44590385 Ki = 2506 nM T36059 C4ORH5 44590386 Ki = 4209 nM T36059 C8IAX2 44590388 Ki = 926 nM T36059 CJT42W 44590830 Ki = 3033 nM T36059 C54CSB 44590831 Ki = 4686 nM T36059 CWM48B 44590832 Ki = 2290 nM T36059 CX98IZ 44590914 Ki = 3047 nM T36059 CDJ76M 44590915 Ki = 1637 nM T36059 CSV95J 44590917 Ki = 5303 nM T36059 CTU78L 44590964 Ki = 5812 nM T36059 CJRT46 44590965 Ki = 410 nM T36059 CU31IQ 44590966 Ki = 5338 nM T36059 C0ZJW7 44590967 Ki = 3547 nM T36059 CQ6Y4N 44593388 Ki = 5288 nM T36059 CZL3S9 44597752 Ki = 17.2 nM T36059 CVW37M 44597868 Ki = 4.9 nM T36059 CV4TA7 44597869 Ki = 4.9 nM T36059 C5KTS9 44597870 Ki = 10.7 nM T36059 CUO03D 44597871 Ki = 120 nM T36059 C1LIA5 44597978 Ki = 404 nM T36059 CM43HO 44598050 Ki = 3640 nM T36059 CC80EX 44598052 Ki = 3450 nM T36059 CYOT49 44598834 Ki = 0.3311 nM T36059 C5ZLC3 44598835 Ki = 0.4266 nM T36059 C6LXZ8 44598836 Ki = 0.3981 nM T36059 CFIA83 44631910 IC50 > 10000 nM T36059 CK05TD 45106502 Ki = 3162.28 nM T36059 CLB20G 45266415 Ki > 100000 nM T36059 CU84YS 45266426 Ki = 29700 nM T36059 CHK6Z9 45267243 Ki = 59 nM T36059 CJZ29E 45267454 Ki = 290 nM T36059 C24KLI 45267987 Ki = 857 nM T36059 CG7M5U 45267990 Ki = 414 nM T36059 C35COL 45267991 Ki = 933.25 nM T36059 C5ZFY1 45268103 Ki = 76.1 nM T36059 CW5TA3 45268108 Ki = 284 nM T36059 CSGE26 45268313 Ki = 209 nM T36059 C7T3HW 45268867 Ki = 707.95 nM T36059 C1IL3E 45268869 Ki = 507 nM T36059 C0OZG5 45268976 Ki = 70.1 nM T36059 C1YSN9 45269707 Ki = 2511.89 nM T36059 C57YDT 45269835 Ki = 90.2 nM T36059 C5H2WJ 45269836 Ki = 37.5 nM T36059 C0Q7RF 45269838 Ki = 75 nM T36059 CJP69G 45270541 Ki = 1063 nM T36059 CTL27N 45271361 Ki = 954.99 nM T36059 CK52VZ 45271363 Ki = 95.5 nM T36059 C20RJQ 45271709 Ki = 16.8 nM T36059 C48IEM 45272391 Ki = 537 nM T36059 CS4L5G 45273118 Ki = 208.93 nM T36059 C6O8XQ 45273122 Ki = 1848 nM T36059 CPG3L9 45481619 Ki = 273 nM T36059 CV13SH 45481620 Ki = 4481 nM T36059 C2ZI4P 45481621 Ki = 1.2 nM T36059 CK2YO1 45481748 Ki = 0.48 nM T36059 CCMX92 45481749 Ki = 36.3 nM T36059 CXM9F4 45481750 Ki = 0.25 nM T36059 CBOG84 45481751 Ki = 11.2 nM T36059 CLZV08 45481752 Ki = 5.86 nM T36059 C3MPR1 45481753 Ki = 1.94 nM T36059 CB52VK 45481754 Ki = 0.93 nM T36059 C5W4NR 45481755 Ki = 330 nM T36059 CQOB79 45481756 Ki = 765 nM T36059 CB8NA2 45481757 Ki = 196 nM T36059 CL68UB 45481758 Ki = 1.25 nM T36059 CY2WO6 45481759 Ki = 268 nM T36059 CV43FT 45481760 Ki = 6.49 nM T36059 C50HVN 45481761 Ki = 125 nM T36059 C4C0QV 45481762 Ki = 65.4 nM T36059 C16LEJ 45481763 Ki = 12.7 nM T36059 C1TB7C 45481764 Ki = 726 nM T36059 CP02LD 45481765 Ki = 3.05 nM T36059 C0L9GH 45481766 Ki = 14.2 nM T36059 CH54CA 45481767 Ki = 0.95 nM T36059 C7GF4H 45481768 Ki = 409 nM T36059 C1FA8U 45481769 Ki = 14.5 nM T36059 C2TWL7 45481770 Ki = 180 nM T36059 C5H7SZ 45481771 Ki = 189 nM T36059 CE80TZ 45482062 Ki = 25 nM T36059 CJG6E4 45482063 Ki = 2306 nM T36059 CVH1A9 45482064 Ki = 71 nM T36059 CGDC50 45482065 Ki = 16 nM T36059 CLRE36 45482066 Ki = 3251 nM T36059 CC3V0B 45482067 Ki = 0.98 nM T36059 C78IES 45482068 Ki = 308 nM T36059 CO96QB 45482069 Ki = 540 nM T36059 CDA2V1 45482070 Ki = 174 nM T36059 CQN78H 45482071 Ki = 692 nM T36059 CF9YU6 45482072 Ki = 359 nM T36059 C9FXY5 45482073 Ki = 120 nM T36059 C12JUY 45482074 Ki = 110 nM T36059 C0FG6J 45482075 Ki = 17.3 nM T36059 CQ5ZF6 45482076 Ki = 0.97 nM T36059 CMI3P8 45482077 Ki = 58.5 nM T36059 CDSG82 45482078 Ki = 12.6 nM T36059 C01FXN 45482079 Ki = 30.5 nM T36059 CE3TD2 45482080 Ki = 95.9 nM T36059 C0IT6Y 45482081 Ki = 207 nM T36059 C0RN6K 45482082 Ki = 100 nM T36059 CD6I4G 45482083 Ki = 1.22 nM T36059 CZ30JX 45482084 Ki = 717 nM T36059 CY49LO 45482085 Ki = 99.8 nM T36059 C1VEW8 45482086 Ki = 189 nM T36059 C8Q6KD 45482087 Ki = 44.4 nM T36059 CP5LN6 45482088 Ki = 223 nM T36059 C12UZF 45482089 Ki = 400 nM T36059 CIF06H 45482090 Ki = 56.5 nM T36059 CDK76E 45482091 Ki = 601 nM T36059 CC52GU 45482092 Ki = 410 nM T36059 CL39ZH 45482093 Ki = 3.47 nM T36059 C8PQ9W 45482094 Ki = 273 nM T36059 COL2R3 45482462 Ki = 5.26 nM T36059 CNDA49 45482464 Ki = 116 nM T36059 CLZM60 45482470 Ki > 10000 nM T36059 CS1L8N 45482471 Ki > 10000 nM T36059 CPX3O6 45482472 Ki > 10000 nM T36059 CZ89HK 45482473 Ki > 10000 nM T36059 CHV46U 45482474 Ki > 10000 nM T36059 C14WOG 45482475 Ki > 1000 nM T36059 CNCK39 45482609 Ki = 61.1 nM T36059 C8JMG7 45482870 Ki = 2.5 nM T36059 C64KXS 45482874 Ki = 0.33 nM T36059 CH4O5W 45483954 Ki = 2.4 nM T36059 C76YLH 45483955 Ki = 0.29 nM T36059 C5Z7IH 45483956 Ki = 12.4 nM T36059 CRT96P 45483957 Ki = 5.5 nM T36059 CNP07M 45483958 Ki = 1.17 nM T36059 CNYS32 45483959 Ki = 11.1 nM T36059 C8PFI3 45483960 Ki = 2.5 nM T36059 CXP5T3 45483961 Ki = 2.17 nM T36059 C48EWA 45483962 Ki = 3.4 nM T36059 CM08CA 45483963 Ki = 3.1 nM T36059 COT4E6 45483964 Ki = 2.1 nM T36059 CG50QU 45483965 Ki = 15.4 nM T36059 C50JZC 45483966 IC50 = 2.5 nM T36059 C7RU6C 45483967 Ki = 57.7 nM T36059 CU6XT8 45483968 IC50 = 1.09 nM T36059 C5BE2O 45483970 Ki = 5270 nM T36059 CX8VT5 45483972 Ki = 4630 nM T36059 C5SR9A 45484443 Ki = 6990 nM T36059 C1J0PG 45484463 Ki = 1720 nM T36059 C8VB0K 45484487 Ki = 10400 nM T36059 CKFZ68 45484498 Ki = 1810 nM T36059 CXVN92 45484506 Ki = 1330 nM T36059 CRE07N 46205479 Ki = 75 nM T36059 C5CV8H 46205480 Ki = 31.4 nM T36059 C5GM2E 46205481 Ki = 72.4 nM T36059 C7YD4H 46205482 Ki = 38.6 nM T36059 C1MS4I 46205483 Ki = 16.7 nM T36059 CG60ME 46205484 Ki = 655 nM T36059 C4B5NU 46205485 Ki = 565 nM T36059 CQK0G9 46205805 Ki = 68.7 nM T36059 CLW1U9 46205806 Ki = 50.6 nM T36059 CRS91E 46205807 Ki = 79.7 nM T36059 CT8E0B 46205808 Ki = 221 nM T36059 C5EZ8J 46205809 Ki = 25 nM T36059 CS3MD6 46205810 Ki = 5 nM T36059 CLAP45 46206128 Ki = 3.43 nM T36059 CK85FB 46206129 Ki = 2.82 nM T36059 CTZ2J4 46206130 Ki = 5.24 nM T36059 CV1HG3 46206131 Ki = 2.1 nM T36059 C0XJ1G 46206132 Ki = 56.4 nM T36059 CT4C0Q 46206133 Ki = 6.88 nM T36059 C9TY8Z 46206464 Ki = 6.94 nM T36059 COIG13 46206465 Ki = 23.9 nM T36059 C5NGI1 46206466 Ki = 153 nM T36059 CYZ9G2 46206467 Ki = 0.108 nM T36059 C8JDB5 46206468 Ki = 0.201 nM T36059 C45TYC 46206469 Ki = 0.248 nM T36059 CHO5B4 46206809 Ki = 0.345 nM T36059 CDS62V 46206810 Ki = 0.241 nM T36059 C7RP3G 46206811 Ki = 0.624 nM T36059 CH34QJ 46226779 Ki = 1.19 nM T36059 C1FO0X 46226780 Ki = 0.97 nM T36059 COZQ07 46226791 Ki = 2.16 nM T36059 CGH6A8 46226792 Ki = 1.35 nM T36059 C3GC7Q 46226793 Ki = 1.04 nM T36059 C4SU3Y 46226794 Ki = 1200 nM T36059 CZ4Y1T 46226797 Ki = 0.97 nM T36059 CV5IZ6 46226798 Ki = 15.6 nM T36059 C5TUH7 46226812 Ki = 0.42 nM T36059 C25QHA 46226822 Ki = 3.03 nM T36059 CSR2C5 46226840 Ki = 2.16 nM T36059 C01JNB 46226841 Ki = 1.17 nM T36059 C6T8DC 46226847 Ki = 35.4 nM T36059 CN2W9P 46226848 Ki = 61.1 nM T36059 C6YJ8O 46226855 Ki = 144 nM T36059 CE5S1Z 46226862 Ki = 31 nM T36059 C8GIE9 46226873 Ki = 94.9 nM T36059 C3EQ6T 46226881 Ki = 135 nM T36059 C78UVJ 46226891 Ki = 97 nM T36059 C8X5EL 46227434 Ki = 113 nM T36059 C5AW2S 46227439 Ki = 433 nM T36059 COW1I2 46227440 Ki = 116 nM T36059 C5C0LN 46228971 Ki = 2160 nM T36059 C3BVX2 46228972 Ki > 1000 nM T36059 C1HNW9 46228973 Ki > 1000 nM T36059 CBI5E6 46228988 Ki = 619 nM T36059 C4IN6L 46229273 Ki > 1000 nM T36059 CURG78 46229274 Ki > 1000 nM T36059 CZ9BN5 46229301 Ki > 1000 nM T36059 CEIJ97 46229302 Ki = 98.8 nM T36059 CN38YO 46229322 Ki > 1000 nM T36059 C9YX4P 46229323 Ki > 1000 nM T36059 C1KVY2 46230151 EC50 = 449 nM T36059 C0YIT3 46230236 EC50 = 44 nM T36059 CV45DT 46230237 EC50 = 42 nM T36059 C7EWV0 46230238 EC50 = 139 nM T36059 CT4AE8 46230239 EC50 = 357 nM T36059 C21NRT 46230240 EC50 = 480 nM T36059 C1B9ZU 46230246 EC50 > 10000 nM T36059 C80CWB 46230290 EC50 = 789 nM T36059 CHG01W 46230545 Ki = 23.6 nM T36059 C4W9GM 46230546 Ki = 29.4 nM T36059 CIK7W5 46230547 Ki = 26 nM T36059 CXP30Y 46230548 Ki = 10.6 nM T36059 CVJ3F6 46230549 Ki = 87.1 nM T36059 C5V6GF 46230550 Ki = 180 nM T36059 C89DAQ 46230551 Ki = 37.5 nM T36059 CJO4C3 46230552 Ki = 9.6 nM T36059 COE2I7 46230553 Ki = 22.3 nM T36059 CBRN59 46230554 Ki = 47 nM T36059 C0EF4K 46230555 Ki = 89.5 nM T36059 C0PG7O 46230556 Ki = 6.5 nM T36059 CFTQ93 46230557 Ki = 102 nM T36059 CVW79B 46230558 Ki = 285 nM T36059 C4JA6N 46230559 Ki = 235 nM T36059 CF13JY 46230560 Ki = 416 nM T36059 C1V2OX 46231332 Ki = 36.4 nM T36059 C7HM3Z 46231333 Ki = 57.7 nM T36059 CV87TC 46231334 Ki = 8.8 nM T36059 CM1H7R 46233161 Ki = 117.49 nM T36059 CI1Z4R 46233211 Ki = 134.9 nM T36059 CW54HP 46233214 Ki = 407.38 nM T36059 CT5CF9 46233315 Ki = 812.83 nM T36059 C7Y6IO 46233346 Ki = 630.96 nM T36059 C7LY3J 46233380 Ki = 245.47 nM T36059 C48HIY 46233446 Ki = 93.33 nM T36059 CEXP72 46237805 Ki = 922 nM T36059 C5TRP3 46237926 Ki = 93 nM T36059 C9GM2W 46237927 Ki = 503 nM T36059 CG57HC 46237928 Ki = 0.6 nM T36059 C0Z1AL 46237929 IC50 = 0.061 nM T36059 CCJ09W 46237930 Ki = 5.9 nM T36059 CN36TB 46237931 Ki = 20.9 nM T36059 C7US4A 46237932 Ki = 357.9 nM T36059 CX5RZ3 46238063 Ki = 29.1 nM T36059 CB6P5J 46238064 Ki = 3 nM T36059 C5LKY8 46238065 Ki = 22.1 nM T36059 CM6K9V 46238066 Ki = 3.7 nM T36059 CMD67R 46238067 Ki = 2.9 nM T36059 C9S4VL 46238068 Ki = 2.9 nM T36059 C7DPI4 46238208 Ki = 120.8 nM T36059 CP9QS1 46238209 Ki = 43.7 nM T36059 CI3S2V 46238210 Ki = 45.2 nM T36059 CS4T7D 46238211 Ki = 22.3 nM T36059 CD60TM 46238212 Ki = 36.3 nM T36059 CX6OK2 46238213 Ki > 1000 nM T36059 CAY7J1 46238338 Ki > 1000 nM T36059 C6PQR8 46238339 Ki > 1000 nM T36059 CWS95Q 46238340 Ki > 1000 nM T36059 CW41JP 46238341 Ki > 1000 nM T36059 C71GBF 46861670 Ki = 2.25 nM T36059 CYC93U 46861671 Ki = 4.26 nM T36059 CLH9D6 46861672 Ki = 5.63 nM T36059 CT6WJ4 46865897 Ki = 633 nM T36059 C5QXL9 46866591 Ki = 1337 nM T36059 C8VJ9K 46866592 Ki = 3754 nM T36059 C9LKD1 46874439 Ki = 31 nM T36059 CC81PS 46874456 Ki = 41 nM T36059 C9UQR8 46874468 Ki = 9.73 nM T36059 CAG1C5 46874475 Ki = 7.8 nM T36059 C27LSE 46874524 Ki = 1.1 nM T36059 C6D5VU 46874588 Ki = 0.33 nM T36059 CA2S6O 46875997 Ki = 4.9 nM T36059 C3KI1M 46876409 Ki = 7.2 nM T36059 CC5OH2 46876751 Ki = 8 nM T36059 CC7B4U 46877219 Ki = 17 nM T36059 CY6S3U 46877262 Ki = 35 nM T36059 CT82OL 46877263 Ki = 23 nM T36059 CKUF93 46877269 Ki = 20 nM T36059 CLU0A9 46877270 Ki = 23 nM T36059 C5D2NU 46877277 Ki = 24 nM T36059 CCH83Y 46877278 Ki = 80 nM T36059 CP3RO7 46877284 Ki = 23 nM T36059 CHI72K 46877285 Ki = 9 nM T36059 C3FJZ9 46877286 Ki = 24 nM T36059 CWD63T 46877289 Ki = 10 nM T36059 COJW51 46877298 Ki = 23 nM T36059 C5MB9D 46877311 Ki = 25 nM T36059 CJ6LH9 46877313 Ki = 20 nM T36059 CFV06U 46877320 Ki = 12 nM T36059 C8H2FW 46877321 Ki = 19 nM T36059 C8C6VB 46877325 Ki = 10 nM T36059 C3F5EW 46877333 Ki = 22 nM T36059 CNYJ02 46877335 Ki = 14 nM T36059 C50XUB 46880372 Ki = 617 nM T36059 CZJ2V5 46880373 Ki = 326 nM T36059 CL8UH3 46880375 Ki = 1866 nM T36059 CQ93IM 46880419 Ki = 189 nM T36059 C7P6TS 46880421 Ki = 4851 nM T36059 CH5B6C 46880424 Ki = 6267 nM T36059 COQ7X3 46880474 Ki = 817 nM T36059 C2SM9Q 46880475 Ki = 715 nM T36059 CV10FQ 46880506 Ki = 471 nM T36059 CEV0M1 46885402 Ki = 170 nM T36059 C9I6WP 46885403 Ki = 4200 nM T36059 CFY8H2 46885404 Ki = 2100 nM T36059 C0X4MS 46885471 Ki = 414 nM T36059 C28VME 46885472 Ki = 2200 nM T36059 CCBF03 46885473 Ki = 4400 nM T36059 C1J2ZP 46885474 Ki = 1020 nM T36059 CO3AF2 46885516 Ki = 5200 nM T36059 CUV1X4 46885517 Ki = 2200 nM T36059 C4A0CV 46885518 Ki = 750 nM T36059 CH70LQ 46885547 Ki = 473 nM T36059 CVG1D3 46885548 Ki = 1050 nM T36059 C4TFD0 46885549 Ki = 2700 nM T36059 C7KD6Q 46885550 Ki = 2200 nM T36059 C06IZF 46885551 Ki = 311 nM T36059 CJ1SV9 46885588 Ki = 9600 nM T36059 C5EGF2 46887668 Ki = 9 nM T36059 C0S7BL 46887669 Ki = 45 nM T36059 CA41WQ 46887671 Ki = 9.02 nM T36059 C0TF5V 46887672 Ki = 5.04 nM T36059 CQP3K6 46887673 Ki = 2.22 nM T36059 CK9P0D 46887898 Ki = 316.23 nM T36059 C9PS5C 46888223 Ki = 280 nM T36059 C6NCF2 46888282 Ki = 25000 nM T36059 CR6T2J 46888283 Ki = 30 nM T36059 C2SX3E 46888356 Ki = 70 nM T36059 C7YGA4 46888359 Ki = 2480 nM T36059 CUFE02 46893147 Ki > 1000 nM T36059 C3JCB1 46911060 Ki = 80 nM T36059 C1LP9S 49796904 Ki = 163 nM T36059 C7E4PO 49796905 Ki = 65 nM T36059 CD1R5K 49796906 Ki = 90 nM T36059 CEK75A 49796907 Ki = 80 nM T36059 CJ8CH9 49863226 Ki = 2806 nM T36059 C8WP4Y 49870952 Ki = 11.8 nM T36059 CE9Q3P 49870953 Ki = 13.2 nM T36059 C56KAX 50940906 Ki = 101 nM T36059 CAKE56 50940909 Ki = 47.3 nM T36059 CR4HU5 50940918 Ki = 157 nM T36059 C0OQI7 50940921 Ki = 4435 nM T36059 C1UMB4 50940926 Ki = 279 nM T36059 CTW9D3 50940928 Ki = 127 nM T36059 CHE59F 50940929 Ki = 142 nM T36059 CCD60O 50940932 Ki = 1279 nM T36059 C17WCS 50940941 Ki = 751 nM T36059 C9UI2X 50940946 Ki = 4.4 nM T36059 CB6QE8 50940947 Ki = 126 nM T36059 CQI9F0 50940948 Ki = 3.6 nM T36059 C6CG1L 50940949 Ki = 71.3 nM T36059 C0I3CZ 50940956 Ki = 25.2 nM T36059 CUS54E 50940957 Ki = 16.7 nM T36059 CG5O0N 50940958 Ki = 63.3 nM T36059 CU89GA 50940959 Ki = 23.99 nM T36059 C9LV4F 50940960 Ki = 18.1 nM T36059 CC6B7M 50940961 Ki = 5.37 nM T36059 CIZ5W0 50940962 Ki = 3.3 nM T36059 CGWA52 50940963 Ki = 15.6 nM T36059 CD1U2T 50940964 Ki = 3 nM T36059 CY7J8X 50940965 Ki = 8 nM T36059 CLY1D0 50940966 Ki = 10.1 nM T36059 C13NAI 50940967 Ki = 20.2 nM T36059 C8I7DL 50940969 Ki = 3.6 nM T36059 C0YSE2 50940970 Ki = 43.6 nM T36059 C26DQG 50940971 Ki = 43.9 nM T36059 CZ4WU9 50940972 Ki = 12.1 nM T36059 CGYR73 50940973 Ki = 23.2 nM T36059 C7CH3U 50940974 Ki = 160 nM T36059 CM2C9F 50940975 Ki = 11.3 nM T36059 CJC06P 50940976 Ki = 14.5 nM T36059 CBFL29 50940977 Ki = 46.9 nM T36059 CB5TZ6 50940978 Ki = 6.2 nM T36059 CMF2S3 50940979 Ki = 21.8 nM T36059 C5H8FK 50940980 Ki = 12.6 nM T36059 CW76LB 50940981 Ki = 64.2 nM T36059 C34PGE 50940982 Ki = 59 nM T36059 C9DR5E 50940985 Ki = 133 nM T36059 CEZM81 50940986 Ki = 34.8 nM T36059 CF8ER6 50940987 Ki = 103 nM T36059 C8X1BV 50940988 Ki = 110 nM T36059 CPB75Y 50940989 Ki = 135 nM T36059 C3Z5KO 50940990 Ki = 10.2 nM T36059 CL1E8H 50941003 Ki = 59 nM T36059 C1B7TN 50941005 Ki = 9.9 nM T36059 CLE1G9 50941006 Ki = 23 nM T36059 CF1V2L 50941009 Ki = 12.2 nM T36059 C1JWZ7 50941010 Ki = 57.54 nM T36059 CH2A9M 50941011 Ki = 32.1 nM T36059 CGTS93 50941012 Ki = 15.85 nM T36059 C8JN6S 50941013 Ki = 52.4 nM T36059 CI6R8X 50941014 Ki = 56.3 nM T36059 CUB5G9 51040798 Ki > 10000 nM T36059 C96NLK 51050843 Ki = 1490 nM T36059 CBX3Q5 51050942 Ki = 3100 nM T36059 CG5P0M 51051040 Ki = 1260 nM T36059 CTZ4H6 51051245 Ki = 8490 nM T36059 C8Z0NV 52912216 IC50 > 10000 nM T36059 CQ5AE4 52936297 Ki = 0.776 nM T36059 C5W4EB 52936298 IC50 = 1.15 nM T36059 CZO2A8 52936299 Ki = 274.2 nM T36059 C4EBJ2 52937820 Ki = 1100 nM T36059 CJK50T 52937925 Ki = 178.4 nM T36059 CER5G6 52937928 IC50 = 28 nM T36059 CR73QA 52937929 Ki = 9.75 nM T36059 C09FNL 52937930 Ki = 8.9 nM T36059 CNPD89 52943141 Ki = 4730 nM T36059 CEFW97 52946211 IC50 = 13000 nM T36059 C8Q3UH 52948332 Ki = 7.244 nM T36059 CK6R3J 52949519 Ki = 4940 nM T36059 C50QVP 53262865 Ki = 859 nM T36059 C7KQP6 53316920 Ki = 239.88 nM T36059 C5BXC0 53316923 Ki = 501.19 nM T36059 CZ7CB2 53317521 Ki = 20 nM T36059 C7A9WB 53318714 Ki = 302 nM T36059 CJZ98W 53318744 Ki = 4076 nM T36059 C42HTK 53321200 Ki = 259 nM T36059 CA91KC 53322692 Ki = 900 nM T36059 CCQR92 53326121 Ki = 269.15 nM T36059 CN51SY 53348048 Ki > 10000 nM T36059 CL3P8I 53394567 Ki = 37 nM T36059 CD2X1W 53469443 Ki = 2429 nM T36059 CUO97T 54577823 Ki > 10000 nM T36059 C9LU8J 54580623 Ki = 5320 nM T36059 CT1CO5 54580654 Ki = 1280 nM T36059 CX3Y6L 54581663 Ki = 1320 nM T36059 C5RQJ9 54582654 Ki = 3290 nM T36059 C08HKQ 54583616 Ki > 1000 nM T36059 CSF9W8 54583714 Ki = 302 nM T36059 CP04UN 54584599 Ki = 3970 nM T36059 CKCD81 54585511 Ki = 22500 nM T36059 CUDT28 54587496 Ki = 0.01 nM T36059 CSL08D 54587662 Ki = 8.472 nM T36059 C83VFS 54754508 Ki = 1.33 nM T36059 C40IVD 54768079 Ki > 10000 nM T36059 C1UW4E 54768080 Ki = 1290 nM T36059 C4JA9T 54768112 Ki > 10000 nM T36059 C2JPC3 54768115 Ki = 1670 nM T36059 CL5SE3 54768601 Ki > 10000 nM T36059 C6SYD1 54768602 Ki > 10000 nM T36059 CX9A4R 54768635 Ki > 10000 nM T36059 C3HNS6 54768636 Ki > 10000 nM T36059 C4VTZ0 54852070 Ki = 680 nM T36059 CUBL54 54852112 Ki = 480 nM T36059 CB7T1O 56627882 Ki = 1.8 nM T36059 C6WSF9 56657920 Ki = 304 nM T36059 CD7C2P 56661442 Ki = 11.4 nM T36059 C2FI4U 56661443 Ki = 28.9 nM T36059 CZ6I4O 56662964 Ki = 500 nM T36059 CVLM74 56664888 Ki = 2.1 nM T36059 CPB29Y 56664889 Ki = 0.2 nM T36059 CBQS24 56668308 Ki = 17.1 nM T36059 CYNJ53 56668410 Ki = 147 nM T36059 CWM34N 56668411 Ki = 3.44 nM T36059 CSJ34D 56668412 Ki = 5.9 nM T36059 C98FPH 56671922 Ki = 4.06 nM T36059 CD6C0P 56675199 Ki = 2.36 nM T36059 CH8YR5 56675200 Ki = 3.02 nM T36059 CUJ34X 56675201 Ki = 3.34 nM T36059 CW3F6I 56675202 Ki = 45 nM T36059 CK3AZ9 56675297 Ki = 1.71 nM T36059 C58FTQ 56675298 Ki = 2.5 nM T36059 C7TNW9 56675299 Ki = 1.72 nM T36059 CDN69Q 56678498 Ki > 10000 nM T36059 CJ6ND1 56678499 Ki = 0.16 nM T36059 C4PL8U 56678500 Ki = 300 nM T36059 C13UZX 56678638 Ki = 5.3 nM T36059 CM04LK 56678639 Ki = 1.91 nM T36059 CVP0A9 56681843 Ki = 1.95 nM T36059 CJ7PC2 56683341 Ki = 600 nM T36059 C02DIY 56838950 Ki > 1000 nM T36059 COY13J 56924646 Ki > 1000 nM T36059 C86NML 56935713 Ki = 450 nM T36059 CB7I4R 56945639 Ki = 138 nM T36059 CXNG25 56945640 Ki = 570 nM T36059 C2RW6L 56945641 Ki = 150 nM T36059 C9XFM7 56945648 Ki = 130 nM T36059 CCK34B 56945649 Ki = 160 nM T36059 C3WC9H 56945650 Ki = 140 nM T36059 CRWJ23 56945749 Ki = 67 nM T36059 CNLD03 56945750 Ki = 220 nM T36059 C78KWY 56945752 Ki = 150 nM T36059 CD54JK 56945753 Ki = 24 nM T36059 CMP74W 56945754 Ki = 24 nM T36059 C5DT0Z 56945768 Ki = 250 nM T36059 CU4C5D 56945769 Ki = 1460 nM T36059 CR1YL9 56945770 Ki = 790 nM T36059 CPA2Z6 56945771 Ki = 620 nM T36059 C9HK5A 56945866 Ki = 39 nM T36059 CMAO83 56945867 Ki = 218 nM T36059 CY4D9S 56945868 Ki = 31.7 nM T36059 C9J2PL 56945870 Ki = 94.2 nM T36059 CKZE52 56945888 Ki = 220 nM T36059 C9VLJ0 56945889 Ki = 260 nM T36059 CRF5J8 56945890 Ki = 140 nM T36059 CX3W2C 56945891 Ki = 200 nM T36059 CD4ZW9 56945994 Ki = 520 nM T36059 CI0Q2T 56945995 Ki = 830 nM T36059 CR5AJ1 56945996 Ki = 320 nM T36059 CH1JR4 56950235 Ki = 15 nM T36059 CXB8Z6 56951623 Ki > 1000 nM T36059 C9T1XQ 56964459 Ki > 10000 nM T36059 CY1IG3 56964460 Ki = 702 nM T36059 CZ42XV 56964461 Ki = 328 nM T36059 CC50SG 56964576 Ki > 10000 nM T36059 CHR8L5 57325914 Ki > 10000 nM T36059 C7SRT3 57325915 Ki > 10000 nM T36059 CREU79 57328471 Ki = 16600 nM T36059 C8JY3E 57384287 IC50 = 60097 nM T36059 CYSA75 57384288 IC50 = 756 nM T36059 CDN54M 57384289 IC50 = 121 nM T36059 CA63RT 57384543 IC50 = 1390 nM T36059 CW63IC 57384544 IC50 = 1407 nM T36059 CCPY02 57385043 IC50 = 113 nM T36059 CKO3L1 57387337 IC50 = 23 nM T36059 C8X7MO 57387594 IC50 = 8 nM T36059 C6XKL9 57387596 IC50 = 7.04 nM T36059 C7XW0T 57387822 IC50 = 1721 nM T36059 CT1R6Q 57387824 IC50 = 141 nM T36059 C01AHY 57387825 IC50 = 259 nM T36059 CNL3P2 57388054 IC50 = 120 nM T36059 CK7R6O 57388055 IC50 = 33 nM T36059 CMBN74 57388056 IC50 = 149 nM T36059 C1BAX6 57391653 Ki = 241 nM T36059 C45GCN 57391694 Ki = 603 nM T36059 C03HUE 57391695 Ki = 507 nM T36059 CJF61Z 57391696 Ki > 1000 nM T36059 CC3X7G 57393433 Ki = 208 nM T36059 C1B3QM 57393434 Ki > 1000 nM T36059 C8ZX4L 57393435 Ki > 1000 nM T36059 CVO2P8 57395120 Ki = 10 nM T36059 C9VWH7 57395161 Ki = 111 nM T36059 CJM7E8 57395162 Ki = 802 nM T36059 CEQR05 57395163 Ki = 61 nM T36059 CDP13M 57395164 Ki = 110 nM T36059 CSTG21 57396888 Ki = 124 nM T36059 CWX64M 57396935 Ki = 749 nM T36059 CC52TB 57396936 Ki = 432 nM T36059 C1WT0H 57396937 Ki > 1000 nM T36059 CD6JT5 57398641 Ki = 55 nM T36059 CHC8U6 57398676 Ki = 526 nM T36059 C1J3DG 57400352 Ki = 83 nM T36059 CNRY34 57400353 Ki = 50 nM T36059 CIX58U 57402117 Ki = 50 nM T36059 CLCX61 57402118 Ki = 12 nM T36059 CBMP08 57402160 Ki = 13 nM T36059 C58APE 57402161 Ki = 125 nM T36059 CKB51R 57402162 Ki = 314 nM T36059 CQK46U 57402163 Ki = 815 nM T36059 CYHD10 57403904 Ki = 161 nM T36059 CD2NO5 57403905 Ki = 315 nM T36059 CR7DG5 57523211 Ki = 1.92 nM T36059 CX1S2Q 57523212 Ki = 4.45 nM T36059 C4IQ0H 57523214 Ki = 2.27 nM T36059 COG52F 57523215 Ki = 6.75 nM T36059 C3LU5I 57523251 EC50 = 0.2512 nM T36059 CQAW53 57523252 EC50 = 12.59 nM T36059 CX0HB3 57523253 EC50 = 19.95 nM T36059 C7SZY3 57523625 Ki = 0.85 nM T36059 C8XE3W 57523626 Ki = 1.01 nM T36059 CV9QD2 57523627 Ki = 0.97 nM T36059 CV13XB 57523628 Ki = 0.97 nM T36059 CO0AH7 57523653 Ki = 0.53 nM T36059 CRXS39 57523654 Ki = 0.58 nM T36059 CR78ZP 57523655 Ki = 1.6 nM T36059 CZTV13 57523656 Ki = 1.22 nM T36059 C5YGB2 57523657 Ki = 0.91 nM T36059 CO2V0F 57523658 Ki = 1.07 nM T36059 CHU5T7 57523687 Ki = 1.65 nM T36059 CWN3A5 57523688 Ki = 1.66 nM T36059 CUSH70 57523689 Ki = 3.78 nM T36059 C5VCS6 57523690 Ki = 10.1 nM T36059 CP9JX0 57523691 Ki = 2.57 nM T36059 CWDV59 57523711 Ki = 3.1 nM T36059 CZIQ36 57523712 Ki = 1.67 nM T36059 CH2KX7 57523713 Ki = 3.48 nM T36059 CO2UQ5 57523714 EC50 = 0.1995 nM T36059 C2U7SP 57523715 Ki = 2.16 nM T36059 C7F4QX 57524978 Ki = 11.1 nM T36059 C4GZY7 58739995 Ki = 444 nM T36059 C1HU4O 59011969 Ki = 7330 nM T36059 CK7T6D 59179887 IC50 > 1000 nM T36059 C5G2RH 60154738 Ki = 25 nM T36059 C4U7BI 60154739 Ki = 3.9 nM T36059 CU3R2Q 60154740 Ki = 10.4 nM T36059 CJ57XU 60154742 Ki = 21 nM T36059 CUK15D 60154835 Ki = 31 nM T36059 CK7VH4 60154837 Ki = 9.7 nM T36059 C3PO4T 60155712 Ki = 65 nM T36059 CJB03P 60155713 Ki = 253 nM T36059 C6W8XE 60155714 Ki = 71 nM T36059 CN03ZC 60155715 Ki = 51 nM T36059 CEZ4V5 60155716 Ki = 25 nM T36059 C1ZXO7 60155796 Ki = 30 nM T36059 CZRU45 60155797 Ki = 24 nM T36059 C8GZ3V 60155798 Ki = 26 nM T36059 CXLO10 60155799 Ki = 13.8 nM T36059 CYB1L4 60155893 Ki = 13.3 nM T36059 C0B5OZ 60155894 Ki = 11.8 nM T36059 CB9A6F 60155895 Ki = 12.4 nM T36059 C2VPM8 60155896 Ki = 44 nM T36059 CW7R1L 60155897 Ki = 39 nM T36059 CP3H2Z 60156002 Ki = 12.2 nM T36059 C8KU5V 60156003 Ki = 30 nM T36059 C2LN4J 60156004 Ki = 9.8 nM T36059 C8SZE0 60156005 Ki = 9.3 nM T36059 CGL84Y 60156006 Ki = 13.7 nM T36059 CFBG07 60156104 Ki = 7.7 nM T36059 CKVJ21 60156105 Ki = 8.1 nM T36059 C7L1BF 60156106 Ki = 6.8 nM T36059 C38NUA 60156107 Ki = 14.5 nM T36059 C87SMR 60156108 Ki = 4.9 nM T36059 C16CSN 60195998 Ki = 1300 nM T36059 C0L8HB 67192741 IC50 = 430 nM T36059 C17YBH 68148396 Ki > 10000 nM T36059 C17JAZ 68284084 IC50 = 8800 nM T36059 C0P1OR 69427076 Ki = 0.76 nM T36059 CXUB67 69846372 Ki = 105 nM T36059 C76KTS 69846756 Ki = 2640 nM T36059 CCDH27 69961639 Ki = 554 nM T36059 C1Q3ST 70676457 Ki = 670 nM T36059 CJ7Y1S 70676459 Ki = 150 nM T36059 COVC42 70676460 Ki = 780 nM T36059 C9OLG0 70676461 Ki = 780 nM T36059 CCO40K 70676610 Ki = 1720 nM T36059 C21ANJ 70676611 Ki = 2930 nM T36059 CN38XM 70676612 Ki = 2790 nM T36059 CYTH16 70676613 Ki = 1760 nM T36059 C0VI8J 70676614 Ki = 550 nM T36059 C5ETD9 70676615 Ki = 790 nM T36059 CJ3PU2 70676773 Ki = 2200 nM T36059 CL04EV 70677099 Ki = 17 nM T36059 CZA8H7 70677100 Ki = 182 nM T36059 C46HBT 70681087 Ki = 560 nM T36059 CIT56B 70681088 Ki = 52 nM T36059 C5W7QI 70681089 Ki = 41.5 nM T36059 CI28FM 70681090 Ki = 83.2 nM T36059 CE3N0Y 70681091 Ki = 40.4 nM T36059 C4ND7L 70682887 Ki = 210 nM T36059 C6FY4R 70682888 Ki = 340 nM T36059 CS0I7Z 70682890 Ki = 0.97 nM T36059 CUP3G0 70684947 Ki = 13 nM T36059 CH83CQ 70684948 Ki = 1320 nM T36059 C0XG9F 70685288 Ki = 500 nM T36059 CK75QB 70685289 Ki = 32.4 nM T36059 CTQ61B 70685290 Ki = 110 nM T36059 CWE50T 70685291 Ki = 114 nM T36059 CWYJ62 70687114 Ki = 8.52 nM T36059 CB4VD0 70687115 Ki = 70 nM T36059 C63KJG 70687116 Ki = 37 nM T36059 CNFS49 70687117 Ki = 140 nM T36059 CM03SU 70687435 Ki = 5.9 nM T36059 CL63IQ 70687436 Ki = 8.9 nM T36059 CWC6O5 70687437 Ki = 16.5 nM T36059 CKY8S0 70689193 Ki = 5.48 nM T36059 C6TVZ8 70689194 Ki = 5.8 nM T36059 CJGO68 70689195 Ki = 200 nM T36059 C1KJD5 70689262 Ki = 100 nM T36059 C7X1UJ 70689496 Ki = 160 nM T36059 C4U2AE 70689497 Ki = 1530 nM T36059 CPI5W0 70689498 Ki = 10.3 nM T36059 CZ9S6P 70691273 Ki = 39 nM T36059 CX2Z3F 70691274 Ki = 54 nM T36059 CTDO23 70691275 Ki = 260 nM T36059 C58QIA 70691614 Ki = 236 nM T36059 C9S1XC 70693389 Ki = 3.2 nM T36059 C3SP8W 70693390 Ki = 100 nM T36059 CDP9H6 70693700 Ki = 6.6 nM T36059 C1KHZ2 70694510 Ki > 10000 nM T36059 CCOX15 70695495 Ki = 5.02 nM T36059 CGW8U4 70695809 Ki = 12.1 nM T36059 CL3E6M 70695810 Ki = 315 nM T36059 C26LVT 70695811 Ki = 12 nM T36059 CVU08A 70695812 Ki = 470 nM T36059 CM1O5S 70695813 Ki = 15.2 nM T36059 C7USK0 70696572 Ki > 1000 nM T36059 CF8V3G 70697511 Ki = 20 nM T36059 CBN9A8 70697521 Ki = 2.3 nM T36059 CAR92Q 71364275 Ki = 75 nM T36059 C31FGM 71412032 Ki = 25 nM T36059 C4O3XF 71449066 Ki = 2.9 nM T36059 CBZM95 71449068 Ki = 14.6 nM T36059 CQCR81 71449139 Ki = 9.8 nM T36059 CXZ40U 71450227 Ki = 404 nM T36059 C38UKP 71450240 Ki = 367 nM T36059 CXM83Y 71450241 Ki = 63.4 nM T36059 C9G0FP 71450242 Ki = 15.4 nM T36059 CC73UY 71450243 Ki = 15.5 nM T36059 CUC9J8 71450828 Ki = 30600 nM T36059 C2PA9L 71450842 Ki = 62500 nM T36059 CTYM41 71450845 Ki = 2.4 nM T36059 C37NIO 71450846 Ki = 11 nM T36059 CW75JC 71450849 Ki = 13.1 nM T36059 C4VMP7 71451329 Ki > 10000 nM T36059 CPQ4Y9 71451659 Ki = 490 nM T36059 C4LVT1 71452054 Ki = 38.1 nM T36059 CC2Q9H 71452055 Ki = 32.7 nM T36059 CQ4CA3 71452056 Ki = 0.3 nM T36059 CWOB13 71452072 Ki = 8.62 nM T36059 CX52PV 71452672 Ki = 0.56 nM T36059 C0MD9G 71452718 Ki = 676 nM T36059 C85LPW 71452749 Ki = 12 nM T36059 C79HWL 71452750 Ki = 35.8 nM T36059 CXF65C 71452801 Ki = 44 nM T36059 C0NC4G 71453140 Ki > 10000 nM T36059 C9QD3W 71453871 Ki = 536 nM T36059 CKW2G6 71453872 Ki = 1360 nM T36059 C0VK4E 71453873 Ki = 35.5 nM T36059 CR8A0V 71453874 Ki = 2.49 nM T36059 CV0NW6 71453875 Ki = 14.9 nM T36059 C5S3FU 71453891 Ki = 241 nM T36059 C0M9CP 71453892 Ki = 44.4 nM T36059 CY1B4N 71453893 Ki = 130 nM T36059 C76PJS 71453894 Ki = 8.57 nM T36059 C43IWS 71453989 IC50 = 850 nM T36059 CO02WB 71454439 Ki = 3.7 nM T36059 C4FBN7 71454511 Ki = 22 nM T36059 C56VEI 71455599 Ki = 156 nM T36059 C79IVN 71455600 Ki = 246 nM T36059 CM2ZF9 71455601 Ki = 38.6 nM T36059 CEO64T 71455602 Ki = 394 nM T36059 CPN0B7 71455603 Ki = 1.07 nM T36059 CUE71P 71455604 Ki = 6.92 nM T36059 CC1RD4 71455619 Ki = 37.6 nM T36059 C2ITP7 71455620 Ki = 37.8 nM T36059 CQ8U5S 71455621 Ki = 5.93 nM T36059 CB2E9C 71455622 Ki = 14.6 nM T36059 CTH1W7 71455623 Ki = 3.82 nM T36059 C1QLP9 71455624 Ki = 17.6 nM T36059 CVJZ12 71456194 Ki = 1.4 nM T36059 CJBC05 71456195 Ki = 0.78 nM T36059 CKU1O4 71456259 Ki = 719 nM T36059 CIE1Z5 71456490 Ki = 6300 nM T36059 C5BHA3 71457388 Ki = 252 nM T36059 CYTZ37 71457389 Ki = 404 nM T36059 C3H2QF 71457390 Ki = 3.71 nM T36059 CPBO67 71457391 Ki = 1.99 nM T36059 C12PEI 71457403 Ki = 309 nM T36059 C19MUP 71457404 Ki = 34.1 nM T36059 CS6Z4N 71457405 Ki = 5.23 nM T36059 C5RD0O 71457406 Ki = 23.8 nM T36059 C6MF5O 71457407 Ki = 7.68 nM T36059 CJA6M2 71457990 Ki = 1.5 nM T36059 C0DPK5 71457992 Ki = 1.6 nM T36059 C6QJ9D 71458047 Ki = 74 nM T36059 C9PG8A 71458089 Ki = 82.9 nM T36059 C5MR7O 71458343 Ki = 5900 nM T36059 CU0YQ6 71459244 Ki = 0.83 nM T36059 CV3L0D 71459245 Ki = 514 nM T36059 CDW92B 71459246 Ki = 36.7 nM T36059 C5WX8S 71459247 Ki = 18 nM T36059 CN79LY 71459248 Ki = 37.8 nM T36059 C82QUK 71459249 Ki = 18.8 nM T36059 CC9I6G 71459250 Ki = 21.1 nM T36059 CQ7BP5 71459268 Ki = 30.9 nM T36059 CG8MI3 71459899 Ki = 0.63 nM T36059 CUI7X3 71459958 Ki = 2280 nM T36059 CA3UR2 71459960 Ki = 163 nM T36059 C8AY0D 71460344 Ki > 10000 nM T36059 CY0LV4 71460666 Ki = 70 nM T36059 CJ1R3V 71460667 Ki = 640 nM T36059 CB9A8S 71461026 Ki = 136 nM T36059 C60OEP 71461027 Ki = 824 nM T36059 CUDN57 71461028 Ki = 4.93 nM T36059 CJ9K0H 71461029 Ki = 187 nM T36059 CDX9O4 71461045 Ki = 822 nM T36059 COU59X 71461116 Ki = 1.9 nM T36059 CA1TQ7 71461609 Ki = 14 nM T36059 C1W0GC 71461630 Ki = 1700 nM T36059 CM6XA5 71461669 Ki = 216 nM T36059 CQ7V9L 71461900 Ki = 4600 nM T36059 CA0EJ2 71462751 Ki = 1330 nM T36059 CK7OB3 71462752 Ki = 356 nM T36059 CP07FL 71462753 Ki = 62.9 nM T36059 CK97MP 71462754 Ki = 96.3 nM T36059 CV1QN8 71462755 Ki = 52.8 nM T36059 COU6E4 71462772 Ki = 182 nM T36059 CGC23V 71462773 Ki = 11 nM T36059 C1HAS6 71462774 Ki = 69.3 nM T36059 CHT04N 71462775 Ki = 47.3 nM T36059 CCZI56 71508483 Ki = 520 nM T36059 C79QVF 71508699 Ki > 1000 nM T36059 CLDQ30 71508726 Ki > 1000 nM T36059 CR3MC4 71508757 Ki > 1000 nM T36059 CCYK35 71508758 Ki > 1000 nM T36059 CCJN86 71511630 Ki = 16.2 nM T36059 CNKZ09 71528098 Ki = 3930 nM T36059 CT29GM 71570217 Ki = 2.8 nM T36059 C79HVM 71570218 Ki = 389 nM T36059 CVY17G 71570219 Ki = 39.81 nM T36059 CFOJ85 71570365 Ki = 512.86 nM T36059 CKGR23 71570366 Ki = 42.4 nM T36059 CBVF69 71570367 Ki = 6.3 nM T36059 CPA1D2 71570369 Ki = 5.2 nM T36059 CLM70H 71570370 Ki = 54.95 nM T36059 CZ4OX3 71570517 Ki = 26.1 nM T36059 CTVU96 71600100 Ki = 75 nM T36059 C69VPU 71601783 Ki = 75 nM T36059 C23UTC 71601785 Ki = 300 nM T36059 C3E6FV 71601786 Ki = 5.6 nM T36059 C5M0ED 71601787 Ki = 2.4 nM T36059 CE89VB 71601788 Ki = 120 nM T36059 CI2T1R 71601789 Ki = 20 nM T36059 CIG9A4 71601928 Ki = 5.3 nM T36059 C0M1JK 71601929 Ki = 5.2 nM T36059 CS02PR 71601930 Ki = 32 nM T36059 C4I6RX 71601931 Ki = 20 nM T36059 C69WKY 71601932 Ki = 7.3 nM T36059 CZ06YT 71601933 Ki = 18 nM T36059 CUB6F0 71602062 Ki = 24 nM T36059 COL4H9 71602063 Ki = 3.2 nM T36059 CN7B9W 71602064 Ki = 25 nM T36059 C7GH1Y 71602065 Ki = 100 nM T36059 C4GEQ0 71602066 Ki = 35 nM T36059 CT0N9X 71602067 Ki = 520 nM T36059 C12CAE 71602199 Ki = 45 nM T36059 CJ8I4C 71602200 Ki = 98 nM T36059 C9T1OI 71602201 Ki = 18 nM T36059 CLZ7U2 71602202 Ki = 24 nM T36059 C81YMF 71602203 Ki = 33 nM T36059 CD0IT5 71602204 Ki = 33 nM T36059 CM87NU 71623050 Ki = 6.4 nM T36059 CNZ17D 71657835 EC50 = 794.33 nM T36059 C70SIG 71680729 Ki > 1000 nM T36059 C0YW1C 71680730 Ki > 1000 nM T36059 CG6EY1 71680731 Ki > 1000 nM T36059 CN0WU1 71680732 Ki > 1000 nM T36059 CK2Y6A 71680733 Ki > 1000 nM T36059 CH5KU9 71680734 Ki = 382 nM T36059 C6OXR9 71680735 Ki > 1000 nM T36059 CA50LT 71680889 Ki > 1000 nM T36059 CCM92I 71680890 Ki = 158 nM T36059 CS51FY 71680891 Ki = 115 nM T36059 CX4BZ6 71680892 Ki > 1000 nM T36059 CC7MA1 71680893 Ki > 1000 nM T36059 C6HZ4O 71680894 Ki > 1000 nM T36059 CN0EZ6 71680895 Ki > 1000 nM T36059 C30NCG 71681049 Ki > 1000 nM T36059 C2TR7P 71681050 Ki > 1000 nM T36059 CVY85K 71681051 Ki = 147 nM T36059 C8TCR6 71681052 Ki > 1000 nM T36059 C4KB8W 71681053 Ki > 1000 nM T36059 CLBD58 71681054 Ki = 91.6 nM T36059 C50TBU 71681055 Ki > 1000 nM T36059 C2Y3KO 71681203 Ki > 1000 nM T36059 CIM0S3 71681204 Ki > 1000 nM T36059 C21UWV 71683091 Ki = 390 nM T36059 COWX82 71683092 Ki = 173 nM T36059 C9CLQ3 71683093 Ki > 1000 nM T36059 CV5O0H 71683094 Ki >= 1000 nM T36059 CCJ17F 71683095 Ki > 1000 nM T36059 C3RD0E 71713167 Ki = 14300 nM T36059 C6SD4L 71764235 Ki = 1.9 nM T36059 C9TWP2 71764236 Ki = 30.2 nM T36059 CZ7SW4 71764237 Ki = 1.23 nM T36059 C8WK5O 71764238 Ki = 12.1 nM T36059 C5EMX3 72197342 Ki = 201 nM T36059 C4E0QC 72197343 Ki > 10000 nM T36059 C76ASV 72197513 Ki = 816 nM T36059 CZW4Y0 72197514 Ki = 567 nM T36059 CUL8V0 72197515 Ki = 2470 nM T36059 CXF4U1 72197516 Ki = 1380 nM T36059 C3QYT8 72197517 Ki = 676 nM T36059 C4W8LQ 72197698 Ki > 10000 nM T36059 CY8GU4 72197699 Ki > 10000 nM T36059 C6BUC3 72197700 Ki > 10000 nM T36059 C48QTY 72197701 Ki = 951 nM T36059 C4D8WO 72197702 Ki = 1870 nM T36059 CAY6J2 72197703 Ki = 2040 nM T36059 C6RDT4 72197880 Ki = 9.36 nM T36059 C7XN0S 72197881 Ki = 746 nM T36059 C5J9QH 72197882 Ki = 36600 nM T36059 CB05ET 72197883 Ki = 918 nM T36059 C52QMK 72197884 Ki > 10000 nM T36059 CWH6T3 72548703 IC50 = 0.17 nM T36059 CS81LQ 72696144 Ki > 10000 nM T36059 C3BEM8 72696145 Ki > 10000 nM T36059 C1E4ZD 72696146 Ki > 10000 nM T36059 CQ35NL 72696147 Ki > 10000 nM T36059 CRN4B1 72696148 Ki > 10000 nM T36059 C0IF1J 72696149 Ki > 10000 nM T36059 CL2H7Y 72696273 Ki > 1000 nM T36059 C7MX9Y 72696274 Ki > 300 nM T36059 CBTE63 72696275 Ki > 10000 nM T36059 CPI89R 72696276 Ki > 10000 nM T36059 COX4B1 72696277 Ki > 10000 nM T36059 CI9HP7 72696397 Ki = 2450 nM T36059 C1RFY6 72696398 Ki = 762 nM T36059 CY56RG 72696399 Ki > 1000 nM T36059 C6A8ZF 72696400 Ki = 541 nM T36059 C8ARZ1 72696401 Ki = 1600 nM T36059 CQ4JZ3 72696520 Ki > 1000 nM T36059 C4DN3V 72696521 Ki > 1000 nM T36059 CWG0U4 72697647 Ki > 10000 nM T36059 CH90JS 72697648 Ki > 1000 nM T36059 CPB7K4 72697649 Ki > 10000 nM T36059 C1D7VQ 72697650 Ki > 1000 nM T36059 C81TXZ 72697651 Ki = 1010 nM T36059 CA5BI1 72697652 Ki > 10000 nM T36059 C50SYX 72697785 Ki = 4410 nM T36059 CXPB58 72697786 Ki > 1000 nM T36059 CJ5W1R 72697787 Ki > 1000 nM T36059 C0CJ6R 72697788 Ki > 1000 nM T36059 CY1I8G 72697789 Ki > 10000 nM T36059 CXDT98 72697790 Ki > 1000 nM T36059 CS7VK8 72697791 Ki > 10000 nM T36059 CX69MI 72697928 Ki > 1000 nM T36059 CT2L7J 72697929 Ki > 1000 nM T36059 CEWO96 72697930 Ki > 1000 nM T36059 CNP9S3 72697931 Ki > 10000 nM T36059 C3NR4V 72697932 Ki > 10000 nM T36059 CQ4IE7 72697933 Ki > 10000 nM T36059 CY94KO 72697934 Ki > 100 nM T36059 CO5K1Y 72698079 Ki > 1000 nM T36059 CVB0Y9 72698080 Ki > 10000 nM T36059 CCOP98 72698081 Ki > 1000 nM T36059 C50ZUX 72698082 Ki = 6800 nM T36059 CZG6V9 72698083 Ki = 3030 nM T36059 C97FMG 72698084 Ki = 3410 nM T36059 CH6Z2U 72698223 Ki = 6320 nM T36059 C3QVP5 72698224 Ki > 10000 nM T36059 CBD03K 72698225 Ki > 10000 nM T36059 CST61L 72698226 Ki > 10000 nM T36059 CJ0GB6 72698227 Ki > 1000 nM T36059 CKP9M2 72698228 Ki > 1000 nM T36059 CW83DK 73213196 Ki > 10000 nM T36059 CRO2K8 73345315 Ki = 0.58 nM T36059 CRW73S 73345316 Ki = 3.6 nM T36059 C4WRE1 73346046 Ki = 9549.93 nM T36059 C5AB9Z 73346835 Ki = 0.83 nM T36059 CF1JN5 73347573 Ki = 389.05 nM T36059 CM5B9S 73347862 Ki > 1000 nM T36059 CTJ0U3 73348946 Ki = 2640 nM T36059 CC3Y7G 73348947 Ki = 67 nM T36059 C2PTH6 73349106 Ki = 794.33 nM T36059 CI65VU 73349920 Ki = 0.69 nM T36059 C4C0GK 73349930 Ki = 0.38 nM T36059 CY5K9T 73350674 Ki = 23.99 nM T36059 CHLF98 73350966 Ki > 1000 nM T36059 CE2YB8 73350967 Ki > 1000 nM T36059 CQSX70 73350968 Ki > 1000 nM T36059 C64LUF 73351429 Ki = 217 nM T36059 C5YXO4 73352175 Ki = 56.23 nM T36059 C5H8SI 73352180 Ki = 2398.83 nM T36059 CIH36P 73352882 Ki = 5.3 nM T36059 C35XEH 73352883 Ki = 5.2 nM T36059 C2M8PJ 73353634 Ki = 28.18 nM T36059 C2IG8X 73353638 Ki = 724.44 nM T36059 CW18JX 73355444 Ki > 1000 nM T36059 C4HX2J 73355960 Ki = 3.1 nM T36059 CH6G8N 73356702 Ki = 5623.41 nM T36059 CF8P0A 73356703 Ki = 7244.36 nM T36059 CMS65T 76309882 Ki = 193 nM T36059 CB84HP 76309883 Ki = 37957 nM T36059 C02EBL 76309925 Ki > 100000 nM T36059 CX1H6Y 76310493 Ki > 100000 nM T36059 C9DL1B 76310832 Ki = 4.6 nM T36059 CGPZ23 76310922 Ki = 12 nM T36059 CCX8V6 76311194 EC50 = 1.585 nM T36059 CQLE57 76311197 EC50 = 39.81 nM T36059 CSV43U 76313599 Ki = 20285 nM T36059 CP2TA1 76313600 Ki = 5233 nM T36059 CQ5Z4P 76313639 Ki = 4460 nM T36059 CY8D4J 76313640 Ki > 100000 nM T36059 CB0WN9 76313641 Ki > 10000 nM T36059 C1C3LK 76314155 Ki > 100000 nM T36059 C25LDC 76314450 Ki = 9.38 nM T36059 CEO9I0 76314563 Ki = 9.2 nM T36059 CZX45G 76314797 EC50 = 100 nM T36059 C21BCT 76317721 Ki = 33500 nM T36059 C2K6XR 76317722 Ki = 10300 nM T36059 CY3V7H 76317723 Ki = 6500 nM T36059 CXQY23 76317724 Ki = 6600 nM T36059 CCY8V2 76318040 Ki = 6.51 nM T36059 CX3H8W 76318139 Ki = 6.7 nM T36059 CNVO51 76318140 Ki = 16 nM T36059 CL4JH8 76318403 EC50 = 5.012 nM T36059 C9O4CQ 76320863 Ki = 4260 nM T36059 CKLB89 76320909 Ki = 2300 nM T36059 CL46PW 76321429 Ki > 60000 nM T36059 CWO42D 76321430 Ki = 5000 nM T36059 CFN3M9 76321431 Ki = 10900 nM T36059 CY5TN2 76321753 Ki = 6.82 nM T36059 C4TO0S 76321824 Ki = 4.9 nM T36059 CHCM51 76321825 Ki = 8.6 nM T36059 C5R6OT 76322076 EC50 = 5.012 nM T36059 CK5Z6L 76324475 Ki = 23307 nM T36059 CHWO53 76324476 Ki = 6419 nM T36059 C3CE4B 76324522 Ki > 10000 nM T36059 C6AV9Z 76325026 Ki = 6700 nM T36059 C1JV7S 76325027 Ki = 11400 nM T36059 CQ51JN 76325369 Ki = 2.74 nM T36059 C2DPT3 76325370 Ki > 30 nM T36059 CP4CY1 76325371 Ki = 2.27 nM T36059 C5J4ML 76325372 Ki > 30 nM T36059 COD78V 76325693 EC50 = 630.96 nM T36059 C3FE0S 76325694 EC50 = 125.89 nM T36059 CC67KO 76328082 Ki > 10000 nM T36059 CA0MJ2 76328083 Ki > 30000 nM T36059 C72UFI 76328084 Ki = 3890 nM T36059 CNM0E1 76328596 Ki = 31900 nM T36059 CXTN91 76328597 Ki = 13500 nM T36059 C3TH4J 76328598 Ki = 8600 nM T36059 CQI9X5 76328599 Ki = 2800 nM T36059 C0AE9L 76328600 Ki = 900 nM T36059 C5B0UO 76328910 Ki = 6.89 nM T36059 C5VEJ9 76328911 Ki > 30 nM T36059 C8O5KF 76329263 EC50 = 3.981 nM T36059 C9O0UH 76329264 EC50 = 39.81 nM T36059 CF82DA 76329265 EC50 = 15.85 nM T36059 CPVN52 76329266 EC50 = 31.62 nM T36059 CG30CO 76331702 Ki = 790 nM T36059 C6QY2P 76331703 Ki = 906 nM T36059 CFNG34 76331754 Ki = 12100 nM T36059 CMR14L 76331755 Ki > 30000 nM T36059 CQT81A 76332277 Ki > 100000 nM T36059 CH64XC 76332278 Ki = 12800 nM T36059 CQWD47 76332279 Ki = 6600 nM T36059 CJKD34 76332280 Ki = 1500 nM T36059 C1GZ8R 76332281 Ki = 7100 nM T36059 CVT1E3 76332599 Ki > 30 nM T36059 CVS3F8 76332600 Ki > 30 nM T36059 CIF6V7 76332686 EC50 = 27.1 nM T36059 CZ27KW 76332687 Ki = 7.8 nM T36059 CYK39X 76332918 EC50 = 2511.89 nM T36059 C4S8NF 76332919 EC50 = 5.012 nM T36059 CF68KC 76335303 Ki = 4300 nM T36059 CL83MV 76335304 Ki = 1952 nM T36059 C7KY5A 76335305 Ki = 3900 nM T36059 CC5IO4 76335344 Ki = 4940 nM T36059 C7FE5D 76335345 Ki = 1280 nM T36059 CIT36F 76335346 Ki = 18300 nM T36059 CV05FX 76335917 Ki > 60000 nM T36059 CLN8S6 76335918 Ki = 23600 nM T36059 CM0D3G 76335919 Ki > 100000 nM T36059 CO86UR 76335920 Ki = 30300 nM T36059 CESR09 76335921 Ki = 5900 nM T36059 CR85PG 76335922 Ki = 2900 nM T36059 C3HE2N 76335923 Ki = 27100 nM T36059 C5DSC0 76335924 Ki = 1300 nM T36059 C5VM4Q 76336198 Ki > 10 nM T36059 CH9WJ4 76336525 EC50 = 10 nM T36059 CNL62P 76336526 EC50 = 10 nM T36059 C5ZRE9 76336527 EC50 = 0.631 nM T36059 CFWX23 82018566 Ki > 1000 nM T36059 CI4M9P 85706712 Ki = 8500 nM T36059 C5T0FH 91799687 EC50 = 1.46 nM T36059 C4BDY3 101676911 Ki = 91.5 nM T36059 C0ROS7 101874280 Ki = 4.14 nM T36059 C1U9RW 101886899 Ki = 6.5 nM T36059 CIE32T 102143331 Ki = 978 nM T36059 CM89YR 102143332 IC50 = 1560 nM T36059 CPRH91 110171405 Ki = 54 nM T36059 CGBO72 118016229 IC50 > 6700 nM T36059 CB74NK 118707149 Ki = 0.86 nM T36059 CP0H8J 118707150 Ki = 11.2 nM T36059 C7UOD9 118707151 Ki = 1.51 nM T36059 CYC0G4 118707152 Ki = 6.16 nM T36059 CLX43G 118707153 Ki = 17.6 nM T36059 C8QTD9 118707154 Ki = 16.5 nM T36059 C4LG6C 118707227 Ki = 11.2 nM T36059 C7W0UA 118707228 Ki = 14.5 nM T36059 CCT74Q 118707229 Ki = 20.2 nM T36059 C8P0JZ 118707230 Ki = 16.9 nM T36059 C6YH5I 118707231 Ki = 4.55 nM T36059 CXD0Y5 118707232 Ki = 8.18 nM T36059 C2ZEU3 118707233 Ki = 7.31 nM T36059 CFH85E 118707843 Ki = 87.7 nM T36059 COX73K 118707844 Ki = 140 nM T36059 CR13GS 118707845 Ki = 730 nM T36059 CS0WC2 118707846 Ki = 18700 nM T36059 C2A3FW 118707847 Ki = 1190 nM T36059 CJ58XH 118707848 Ki = 1350 nM T36059 CF78CL 118707849 Ki = 4220 nM T36059 C3K7UV 118707850 Ki = 553 nM T36059 C0UFO4 118707851 Ki = 357 nM T36059 CSW70B 118707852 Ki = 2510 nM T36059 CU9OE7 118707853 Ki = 2590 nM T36059 CGJW82 118707854 Ki = 59400 nM T36059 CUR32J 118707855 Ki = 3.3 nM T36059 C6O0RY 118707856 Ki = 11.3 nM T36059 CG10IH 118707857 Ki = 9.46 nM T36059 C9OHF2 118707858 Ki = 39.3 nM T36059 CW72CL 118707859 Ki = 9.52 nM T36059 CL0U3C 118707860 Ki = 35 nM T36059 CL3NG5 118707861 Ki = 41.2 nM T36059 C9BSD0 118707862 Ki = 10 nM T36059 CDTJ73 118707863 Ki = 56.1 nM T36059 CRDU39 118707864 Ki = 57.6 nM T36059 C6Y5VQ 118707865 Ki = 46.3 nM T36059 CBO8V9 118707866 Ki = 56.8 nM T36059 C4CU6D 118707867 Ki = 323 nM T36059 C4P5GH 118707868 Ki = 875 nM T36059 C9FKE5 118707869 Ki = 336 nM T36059 CNJ3Z4 118707870 Ki = 11.7 nM T36059 CXQY36 118707871 Ki = 321 nM T36059 C7SL4C 118707872 Ki = 517 nM T36059 CFR3Z1 118707873 Ki = 836 nM T36059 C87ATB 118707874 Ki = 1770 nM T36059 C7HS6T 118707875 Ki = 275 nM T36059 CXHQ82 118707876 Ki = 8700 nM T36059 CEQP75 118707877 Ki = 131 nM T36059 CY8OV1 118707878 Ki > 30000 nM T36059 CH5B6Y 118707879 Ki = 24.4 nM T36059 C3OJW0 118707880 Ki = 1190 nM T36059 CM5BE7 118707881 Ki = 15900 nM T36059 CHR1E9 118707882 Ki = 480 nM T36059 CZW6U4 118707883 Ki = 26300 nM T36059 COR57B 118707884 Ki = 17500 nM T36059 C8C9TQ 118707885 Ki = 16400 nM T36059 C0NQ2O 118707886 Ki = 165 nM T36059 CG68RH 118707887 Ki = 17700 nM T36059 C9CY3P 118707888 Ki = 15800 nM T36059 CNC81J 118707889 Ki = 2230 nM T36059 CM53PE 118707890 Ki = 751 nM T36059 CL4B7K 118707891 Ki = 5520 nM T36059 CR20MO 118707892 Ki = 14000 nM T36059 C8WQ5E 118707893 Ki = 11600 nM T36059 CI6O9D 118707894 Ki = 15900 nM T36059 C28ABD 118707895 Ki = 28300 nM T36059 C56KNQ 118707896 Ki = 2070 nM T36059 C7LNI5 118708213 Ki = 97 nM T36059 CBG4I3 118708219 Ki = 572 nM T36059 C50PKS 118708228 Ki = 435 nM T36059 C7W5XN 118708576 Ki = 560 nM T36059 CYO73E 118714540 Ki = 207 nM T36059 CJEW03 118714541 Ki = 1810 nM T36059 C0N4FO 118714542 Ki = 1960 nM T36059 CQZ6I2 118714543 Ki = 171 nM T36059 CI76CX 118719026 Ki = 2.4 nM T36059 C1DF9H 118721207 Ki = 72 nM T36059 CF32CY 118721208 Ki = 166 nM T36059 CQ7I0M 118721210 Ki = 245 nM T36059 CPXH85 118721212 Ki = 31.9 nM T36059 CR9D2E 118721213 Ki = 12.5 nM T36059 C91QXI 118721214 Ki = 171 nM T36059 CCL9T3 118721215 Ki = 25.1 nM T36059 C3BP7M 118721216 Ki = 39.4 nM T36059 C8STW6 118721217 Ki = 23.3 nM T36059 C7MHX0 118721218 Ki = 54.8 nM T36059 COV9Y2 118721219 Ki = 231.4 nM T36059 CM60VZ 118721483 Ki = 545 nM T36059 CZEL84 118721484 Ki = 15.2 nM T36059 CN4SK2 118721485 Ki = 23.9 nM T36059 CYBW39 118721486 Ki = 26.6 nM T36059 CSO42U 118723504 Ki = 308.4 nM T36059 C1SN3J 118723507 Ki = 64 nM T36059 CZV1B8 118723509 Ki = 193.2 nM T36059 C2NBS8 118729966 Ki = 4120 nM T36059 CBH8G1 118729967 Ki = 8220 nM T36059 CA3IK7 118729968 Ki = 2160 nM T36059 CTL02Y 118729969 Ki = 520 nM T36059 CGTA19 118729970 Ki = 4090 nM T36059 C8KX7U 118729971 Ki = 4710 nM T36059 CWJ48N 118729972 Ki > 30000 nM T36059 CU0W7P 118729973 Ki = 35600 nM T36059 CAS85G 118729974 Ki = 34000 nM T36059 CFX4R9 118729975 Ki = 7130 nM T36059 C6VC5A 118729976 Ki = 334 nM T36059 CNG5S7 118729977 Ki > 10000 nM T36059 CD6GZ2 118729978 Ki = 9560 nM T36059 C03XWO 118729979 Ki = 330 nM T36059 CZD98F 118729980 Ki = 3870 nM T36059 CE5Z7R 118729981 Ki = 2730 nM T36059 CBV0J4 118729982 Ki > 30000 nM T36059 C2A5CU 118729983 Ki = 3910 nM T36059 C5FU1D 118730334 Ki = 0.77 nM T36059 CK1Z8H 118730335 Ki = 0.91 nM T36059 CQX2Z3 118730336 Ki = 0.63 nM T36059 CSX6B1 118730337 Ki = 3.39 nM T36059 CL8Q0E 118730338 Ki = 2.16 nM T36059 CO9BI5 118730339 Ki = 2.15 nM T36059 C2AJP8 118730340 Ki = 2.07 nM T36059 CI9BG8 118730341 Ki = 1.97 nM T36059 C43HRM 118730342 Ki = 3.53 nM T36059 CJ1F2N 118730343 Ki = 2.23 nM T36059 C5ZKW3 118730344 Ki = 2.34 nM T36059 C9HFE1 118730345 Ki = 0.62 nM T36059 C3YGD9 118730346 Ki = 1.45 nM T36059 CI8M9O 118730347 Ki = 1.5 nM T36059 CZ29SU 118730348 Ki = 1.62 nM T36059 C5PN4I 118730349 Ki = 0.52 nM T36059 CI1L8O 118730350 EC50 = 0.42 nM T36059 C6HV3B 118730351 Ki = 0.7 nM T36059 C3LZM9 118730352 Ki = 0.44 nM T36059 CU4GY3 118730353 Ki = 2.1 nM T36059 CI34DV 118730354 Ki = 1.15 nM T36059 C25XKA 118730355 Ki = 1.68 nM T36059 CM3S0N 118732278 Ki > 100000 nM T36059 CWQ54J 118732279 Ki > 100000 nM T36059 CQL0K7 118732280 Ki = 19700 nM T36059 CRK7H9 118732281 Ki = 32900 nM T36059 CK24DH 118732282 Ki = 900 nM T36059 CP78KH 118732283 Ki = 14000 nM T36059 CEO92J 118732284 Ki = 10400 nM T36059 CJ6YF9 118732285 Ki = 18100 nM T36059 CW62JS 118732286 Ki > 100000 nM T36059 CXW9U6 118732287 Ki > 100000 nM T36059 C06FRT 118732288 Ki > 100000 nM T36059 CR2CO8 118732289 Ki = 100000 nM T36059 C94GHE 118732290 Ki = 8600 nM T36059 COJ86X 118732291 Ki = 5700 nM T36059 C1KDT4 118732292 Ki > 100000 nM T36059 C7BO1N 118732293 Ki = 28000 nM T36059 C4EFY5 118732294 Ki = 4300 nM T36059 CKV50L 118732295 Ki = 12200 nM T36059 CT3Q9E 118732296 Ki = 6800 nM T36059 CLRK73 118732297 Ki = 5800 nM T36059 CE85HO 118732298 Ki = 3000 nM T36059 C9Y6EK 118732299 Ki = 3600 nM T36059 CNJ1H0 118732300 Ki = 2200 nM T36059 CX6IN3 118732301 Ki > 100000 nM T36059 C4N6ZT 118732302 Ki = 2900 nM T36059 CDAZ14 118732303 Ki > 100000 nM T36059 CZ7TM6 118732304 Ki = 5400 nM T36059 CXZW46 118732305 Ki > 100000 nM T36059 CWX3P4 118732306 Ki = 14600 nM T36059 CXRT76 118732307 Ki = 13300 nM T36059 CK0NS3 118732308 Ki = 4300 nM T36059 CRFJ71 118732309 Ki = 10400 nM T36059 CT90VA 118732971 Ki = 3.86 nM T36059 CXM53U 118732972 Ki = 0.478 nM T36059 CF4G3P 118732973 Ki = 0.429 nM T36059 C3E2BJ 118732974 Ki = 0.875 nM T36059 C1U2FS 118732975 Ki = 0.461 nM T36059 C4YS5J 118732976 Ki = 8.85 nM T36059 CZ7QU0 118732977 Ki = 16.1 nM T36059 CHP93T 118732978 Ki = 15.4 nM T36059 CBT95M 118732979 Ki = 9.62 nM T36059 CZ3X0P 118732980 Ki = 2.61 nM T36059 CMDH59 118732981 Ki = 4.71 nM T36059 C7MZ9V 118732982 Ki = 0.588 nM T36059 C9OCJ2 118733033 Ki = 384 nM T36059 C4PWI2 118733034 Ki = 826 nM T36059 CXQ9Y8 118733035 Ki = 109 nM T36059 CW08YQ 118733049 Ki = 450 nM T36059 C5O2RV 118733056 Ki = 110 nM T36059 CVS8R0 118734340 Ki = 2161 nM T36059 C91DBT 118734341 Ki = 5502 nM T36059 CV1JE8 118734342 Ki = 3252 nM T36059 C8AB7F 118734343 Ki = 4083 nM T36059 CLWV70 118734344 Ki = 1874 nM T36059 CP7SE9 118734345 Ki = 1677 nM T36059 CC0RE9 118734346 Ki = 1306 nM T36059 CV6X3F 118734347 Ki = 3382 nM T36059 CN8RI9 118734348 Ki = 2034 nM T36059 CEZ86B 118734349 Ki = 759 nM T36059 C1QPJ3 118734350 Ki = 2655 nM T36059 CFH92R 118734351 Ki = 2052 nM T36059 CR8FT9 118734352 Ki = 2195 nM T36059 C8Y7QW 118734353 Ki = 5833 nM T36059 CR3Y1J 118734354 Ki = 5884 nM T36059 C5DL3X 118734355 Ki = 1172 nM T36059 CYB49C 118734356 Ki > 10000 nM T36059 CZE09N 118734357 Ki = 1870 nM T36059 CB7J1G 118734358 Ki = 1387 nM T36059 C79RHZ 118734359 Ki = 3425 nM T36059 CSAH95 118734360 Ki = 1845 nM T36059 C1CBG3 118734361 Ki = 1538 nM T36059 CN9S1Y 118734362 Ki = 764 nM T36059 C5SQA1 118734363 Ki = 1003 nM T36059 CDVO89 118734364 Ki = 1818 nM T36059 CQ73IF 118734365 Ki = 1487 nM T36059 C43VAO 118734366 Ki = 3481 nM T36059 C4NQV6 118734367 Ki > 10000 nM T36059 CGF84C 118734368 Ki > 10000 nM T36059 C94UXF 118734369 Ki = 70 nM T36059 CU0K8H 118734370 Ki = 293 nM T36059 CPY5O0 118734371 Ki = 37 nM T36059 CLI1V7 118734372 Ki = 36 nM T36059 CX08QC 118734373 Ki = 43 nM T36059 CD3BV5 118734374 Ki = 39 nM T36059 C58VBC 118734375 Ki = 248 nM T36059 C0U1NA 118734376 Ki = 62 nM T36059 CZH87J 118734377 Ki = 437 nM T36059 C6R5EX 122178744 Ki = 79 nM T36059 CH7X6K 122178745 Ki = 63 nM T36059 C4EW6R 122178746 Ki = 42 nM T36059 C0ORM6 122178747 Ki = 122 nM T36059 C7WCK3 122178748 Ki = 71 nM T36059 C0V6CM 122178749 Ki = 345 nM T36059 C6CQP9 122178750 Ki = 30 nM T36059 C3Z2FP 122178751 Ki = 18 nM T36059 C1HA2V 122178752 Ki = 155 nM T36059 C4LN2B 122178753 Ki = 89 nM T36059 CC6X3Q 122178754 Ki = 520 nM T36059 CA25IQ 122178755 Ki = 29 nM T36059 CSKN51 122178756 Ki = 33 nM T36059 C79XUV 122178757 Ki > 1000 nM T36059 CRJE23 122185011 IC50 = 370 nM T36059 CYF6J5 122188570 Ki = 3.8 nM T36059 C1CJQ0 122188571 Ki = 1.1 nM T36059 C1V7EC 122188572 Ki = 2.9 nM T36059 C3HUJ5 122188573 Ki = 2.9 nM T36059 COC50K 122188574 Ki = 1 nM T36059 CM1I6S 122188575 Ki = 4.5 nM T36059 CZ38MA 122188576 Ki = 7.9 nM T36059 CI9B1A 122188577 Ki = 15 nM T36059 CI7PV6 122188578 Ki = 3 nM T36059 CHVR64 122188579 EC50 = 1.5 nM T36059 CG98FV 122188580 Ki = 38 nM T36059 CV2EG4 122188581 Ki = 10 nM T36059 C2UIX0 122188582 Ki = 0.73 nM T36059 CKXN74 122188583 Ki = 1.2 nM T36059 C2WK9L 122188584 Ki = 9.4 nM T36059 CHEV48 122188585 Ki = 21 nM T36059 C7D6KI 122188586 Ki = 110 nM T36059 CU8HB2 123131614 Ki = 720 nM T36059 CX43WO 123131616 Ki = 5660 nM T36059 CKW26O 123131618 Ki = 780 nM T36059 C9OR6D 127025959 IC50 = 269.15 nM T36059 CXG31M 127026188 Ki = 985 nM T36059 CS7TW8 127026252 IC50 = 79.43 nM T36059 C0MWD8 127026257 IC50 = 2.291 nM T36059 CQ6ND4 127027224 Ki = 910 nM T36059 C48DKZ 127034217 Ki = 4611 nM T36059 CPDA12 127034814 Ki = 33 nM T36059 CZ61LK 127034966 EC50 > 5011.87 nM T36059 CA0SN5 127034967 EC50 > 5011.87 nM T36059 CHTC74 127034991 Ki = 9.54 nM T36059 CH6L8J 127035004 Ki = 9.7 nM T36059 C2BM4D 127035624 Ki = 170 nM T36059 CFJ95C 127035625 Ki = 349 nM T36059 CPY0S3 127035626 Ki = 29.7 nM T36059 CDWC03 127035803 Ki = 1670 nM T36059 CH41BT 127035804 Ki = 257 nM T36059 C7AHR2 127035805 Ki = 286 nM T36059 C92RXW 127035806 Ki = 45.5 nM T36059 CGD59Y 127035832 Ki = 905 nM T36059 CX29PN 127035833 Ki = 105 nM T36059 C4Y3XI 127035834 Ki = 129 nM T36059 CKO8J5 127036423 Ki = 5.87 nM T36059 CP19FZ 127036424 Ki = 2.12 nM T36059 CJM9Z1 127036437 Ki = 1560 nM T36059 CM63GQ 127036438 Ki = 572 nM T36059 CW64ZN 127036450 Ki = 78 nM T36059 C7GHF9 127036560 Ki = 0.027 nM T36059 CZN8O9 127036561 Ki = 3.53 nM T36059 CA4E7T 127036562 Ki = 2.34 nM T36059 CLI39Z 127036563 Ki = 2.43 nM T36059 COD60T 127036564 Ki = 0.41 nM T36059 C59HYJ 127036640 Ki = 294 nM T36059 CJ52XA 127036641 Ki = 375 nM T36059 CX9H5M 127036642 Ki > 100000 nM T36059 C4F2WP 127036740 Ki = 9240 nM T36059 C3QVM7 127036741 Ki = 13400 nM T36059 C3E7ZT 127036742 Ki = 8500 nM T36059 CGM30I 127036810 Ki = 455 nM T36059 CR7OT4 127036811 Ki = 275 nM T36059 CR58OX 127036812 Ki = 114 nM T36059 C65YKX 127036844 Ki = 37 nM T36059 CLCF05 127036845 Ki = 557 nM T36059 C5K3MR 127036846 Ki = 1300 nM T36059 C01OSA 127036925 Ki = 9.83 nM T36059 CB8HG0 127036933 Ki = 250 nM T36059 C1MS0C 127036976 Ki = 75.3 nM T36059 CQR43P 127036977 Ki = 123 nM T36059 CDH32Z 127037385 Ki = 223 nM T36059 C2G1FL 127037386 Ki = 202 nM T36059 CEG84J 127037422 Ki = 6.42 nM T36059 CE5RO8 127037423 Ki = 1.31 nM T36059 CMF9R6 127037424 Ki = 1.82 nM T36059 CY71PR 127037440 Ki = 250 nM T36059 CR57HS 127037441 Ki = 17 nM T36059 C7LV5T 127038039 Ki = 123 nM T36059 C72DGU 127038339 Ki = 1224 nM T36059 CB5F1H 127038752 Ki = 81 nM T36059 CR3A5Y 127038753 Ki = 121 nM T36059 C2KN6C 127038754 Ki = 40.6 nM T36059 CN2R1H 127038755 Ki = 55.6 nM T36059 C86CAO 127038756 Ki = 228 nM T36059 C5IL3Q 127038757 Ki = 169 nM T36059 CVA6S8 127041419 Ki = 231 nM T36059 CXA76Q 127041420 Ki = 122 nM T36059 CN2R5C 127041421 Ki = 75 nM T36059 C04FIN 127043159 Ki > 1000 nM T36059 CXK89P 127043160 Ki > 1000 nM T36059 CB9Q2K 127043161 Ki > 1000 nM T36059 CD23GH 127043299 Ki = 1460 nM T36059 CAK8N9 127043339 Ki > 1000 nM T36059 C5PBH0 127043340 Ki > 1000 nM T36059 CG8F3I 127043648 Ki = 3420 nM T36059 C93XPB 127043661 Ki > 1000 nM T36059 CZ5BA7 127043662 Ki > 1000 nM T36059 C63QSD 127043663 Ki > 1000 nM T36059 CKG3S7 127043664 Ki = 633 nM T36059 C57BHD 127043668 Ki > 1000 nM T36059 C9JY6M 127043669 Ki = 619 nM T36059 CH8S0Y 127043671 Ki > 1000 nM T36059 CU6I9L 127043672 Ki > 1000 nM T36059 CQVE62 127043673 Ki > 1000 nM T36059 C1J3PR 127043818 Ki = 1290 nM T36059 C8V5EN 127043828 Ki = 310 nM T36059 C1PXL8 127043829 Ki = 890 nM T36059 CN46BI 127043830 Ki > 1000 nM T36059 COW15S 127043831 Ki > 1000 nM T36059 C2HWP1 127043995 Ki > 1000 nM T36059 CMJL86 127044142 Ki = 3190 nM T36059 CYS6Z4 127044283 Ki = 934 nM T36059 CC6MG4 127044514 Ki = 563 nM T36059 CW18JP 127044515 Ki = 843 nM T36059 C4O7WX 127044516 Ki = 3630 nM T36059 C3KQS4 127044517 Ki = 1070 nM T36059 CE1A4H 127044518 Ki = 1280 nM T36059 CQJ71U 127044681 Ki = 8630 nM T36059 CS0M2P 127044784 Ki > 1000 nM T36059 C7V4HX 127044785 Ki = 3900 nM T36059 CLXU52 127044795 Ki = 594 nM T36059 C5FC3T 127044855 Ki = 978 nM T36059 CB35MD 127045017 Ki > 1000 nM T36059 CO9LP5 127045018 Ki > 1000 nM T36059 C87ISU 127045019 Ki > 1000 nM T36059 C8W3FJ 127045020 Ki > 1000 nM T36059 CK0ST8 127045021 Ki > 1000 nM T36059 C53KHG 127045164 Ki = 17200 nM T36059 C5LC0U 127045165 Ki = 2650 nM T36059 CGS9B5 127045166 Ki > 100000 nM T36059 C8NV5Y 127045167 Ki > 1000 nM T36059 C2R9PY 127045168 Ki > 1000 nM T36059 C0RMT7 127045169 Ki > 1000 nM T36059 C7I3NV 127045170 Ki > 1000 nM T36059 CRF57W 127045471 Ki > 1000 nM T36059 CW6B7M 127045472 Ki > 1000 nM T36059 C7FH4S 127045473 Ki > 1000 nM T36059 C9QIC7 127045630 Ki > 1000 nM T36059 C6UK3Q 127045631 Ki > 1000 nM T36059 CQL9K1 127045632 Ki > 1000 nM T36059 C8MT9L 127045699 Ki = 498 nM T36059 C02HYP 127045700 Ki = 427 nM T36059 C6VU1I 127045701 Ki = 71 nM T36059 C2GH3Q 127045815 Ki = 147 nM T36059 CV18FC 127045824 Ki = 150 nM T36059 C4MQU2 127045909 Ki = 122 nM T36059 CQ1IB0 127045910 Ki = 225 nM T36059 CDHL50 127046050 Ki = 88 nM T36059 C80WYL 127046438 Ki = 209 nM T36059 CH8W3C 127046493 Ki = 196 nM T36059 COE1R5 127046494 Ki = 905 nM T36059 C72JQB 127046495 Ki = 269 nM T36059 C9OQ3P 127046496 Ki = 82 nM T36059 C51CEW 127047146 Ki = 297 nM T36059 C6WC1L 127047147 Ki = 375 nM T36059 CAN9C7 127047802 Ki = 163 nM T36059 CW64PN 127047804 Ki = 405 nM T36059 C5XZN0 132007291 Ki = 120 nM T36059 C1TJ7B 132578491 Ki > 10000 nM T36059 C5CKG0 132578492 Ki = 14000 nM T36059 CVS8H1 132578493 Ki >= 10000 nM T36059 CKIA45 132933622 Ki = 6860 nM T36059 CA31YG 132938348 Ki = 0.57 nM T36059 CJ54MF 132991405 Ki = 36 nM T36059 C75XIA 132991406 Ki = 92 nM T36059 C3UC1T 134132667 Ki = 287 nM T36059 C2I7AE 134132684 Ki = 1884 nM T36059 CHSK61 134133787 Ki = 824 nM T36059 CH53WN 134134340 Ki = 2390 nM T36059 CR38DS 134138275 Ki = 55 nM T36059 C7WPX1 134138322 Ki = 2652 nM T36059 CV38YZ 134138961 Ki = 381 nM T36059 CIAY28 134139825 Ki = 321 nM T36059 C2KSZ9 134142435 Ki = 35 nM T36059 C5ZAD2 134142611 Ki = 76 nM T36059 CR1YQ6 134142843 Ki = 23600 nM T36059 C5L9BD 134143752 Ki = 236 nM T36059 C3L2PZ 134147788 Ki = 37 nM T36059 CRA5O4 134147994 Ki = 1135 nM T36059 CPI01N 134149255 Ki = 217 nM T36059 CNET28 134151346 Ki = 35 nM T36059 C8PT9W 134152052 Ki = 34 nM T36059 C1JK6T 134152846 Ki = 546 nM T36059 C20RNA 134157761 Ki = 23 nM T36059 C08ZQW 135404340 Ki > 10000 nM T36059 C49ATB 135404761 IC50 = 1.2 nM T36059 CC0P2Z 135405211 IC50 = 0.41 nM T36059 C9WD5K 135405767 Ki = 16 nM T36059 C61NZE 135409562 Ki = 0.2 nM T36059 C2ATW9 135409793 IC50 = 0.67 nM T36059 CRVK68 135409825 Ki = 190 nM T36059 C5T2ZE 135409960 Ki = 27 nM T36059 C4MAB0 135413969 Ki = 22000000 nM T36059 C6G0HA 135416050 Ki > 1000 nM T36059 CI0HT3 135416055 Ki > 1000 nM T36059 C1IEY0 135418256 IC50 = 4.9 nM T36059 C0C5IU 135418454 Ki = 0.61 nM T36059 C0Z8RU 135421343 Ki > 1000 nM T36059 CW16MF 135421366 Ki > 1000 nM T36059 CUA67Z 135423046 Ki = 0.14 nM T36059 CLK7X1 135427226 IC50 = 1 nM T36059 CY9QI4 135428630 Ki > 10000 nM T36059 C7P2ME 135428645 Ki > 10000 nM T36059 C5OZ0L 135428653 Ki > 10000 nM T36059 CI4Z3R 135430228 Ki > 1000 nM T36059 CZA5F9 135436760 Ki > 1000 nM T36059 CJ6AW4 135437132 Ki = 209 nM T36059 CNJ9P7 135437142 IC50 = 1.9 nM T36059 C6HN3Z 135438480 Ki = 521 nM T36059 CI4S7C 135440168 Ki > 1000 nM T36059 CR9W5J 135440414 Ki > 1000 nM T36059 C1UNH9 135440428 Ki > 1000 nM T36059 CXY13D 135440607 IC50 = 0.33 nM T36059 C3JA5S 135442119 Ki = 610 nM T36059 CAG0W3 135442266 IC50 = 1.2 nM T36059 C5YUC2 135443302 Ki > 1000 nM T36059 CO87CV 135443324 Ki > 1000 nM T36059 CWD8M7 135443353 Ki > 1000 nM T36059 C4KLO0 135443378 Ki > 1000 nM T36059 CAO3L2 135443744 IC50 = 0.25 nM T36059 CG9IK2 135444614 IC50 = 0.3 nM T36059 CLY1V5 135447756 IC50 = 0.41 nM T36059 C9UCG0 135448286 Ki > 1000 nM T36059 C7D0AO 135450786 IC50 = 0.3 nM T36059 C0B1XV 135454766 Ki = 27 nM T36059 C4DUN5 135464144 IC50 < 0.1 nM T36059 C2Z0TJ 135465623 IC50 = 1.1 nM T36059 CT4L7M 135465666 Ki = 175 nM T36059 CK47BF 135465712 Ki = 73 nM T36059 CU14JT 135465774 Ki > 1000 nM T36059 C1F5CA 135465776 Ki > 1000 nM T36059 C04XNV 135465778 Ki > 1000 nM T36059 CBV8I2 135465784 Ki > 1000 nM T36059 C7E2CQ 135465796 Ki > 1000 nM T36059 CX04SI 135470376 IC50 = 680 nM T36059 C15FUA 135470377 IC50 = 1.8 nM T36059 C0YZ3B 135470411 Ki > 1000 nM T36059 C5F1TQ 135475602 IC50 = 0.45 nM T36059 CW4V3S 135475677 Ki = 63 nM T36059 CPQ3J6 135477916 Ki = 19 nM T36059 CXJ12O 135479920 IC50 = 0.27 nM T36059 CK52RH 135483531 Ki > 1000 nM T36059 CTU21N 135483619 Ki = 44 nM T36059 CJ91TZ 135484407 IC50 = 4 nM T36059 C7A8ML 135484632 IC50 = 9.1 nM T36059 CI8R0L 135485985 Ki = 348 nM T36059 CE26MK 135486084 Ki > 1000 nM T36059 CH0AR8 135486118 Ki > 1000 nM T36059 C94GIL 135490950 Ki = 90 nM T36059 C2PVW5 135491190 Ki = 28000 nM T36059 CVG5M0 135493238 Ki > 1000 nM T36059 CCX3D7 135493268 Ki > 1000 nM T36059 CF06CK 135493272 Ki > 1000 nM T36059 CS3OC8 135493279 Ki > 1000 nM T36059 C9RS5H 135493280 Ki > 1000 nM T36059 CEI8W7 135493281 Ki > 1000 nM T36059 C25QGD 135493285 Ki > 1000 nM T36059 CN10IO 135493286 Ki > 1000 nM T36059 C7O1NS 135493290 Ki > 1000 nM T36059 CV4X0H 135493292 Ki > 1000 nM T36059 C5OK7A 135499926 Ki > 1000 nM T36059 CG3V6J 135501712 Ki = 179 nM T36059 CQ0W8I 135504131 Ki = 140 nM T36059 CU8W5N 135508372 Ki = 9 nM T36059 C28UOK 135509755 Ki = 140 nM T36059 CHM19U 135512719 IC50 = 610 nM T36059 C89IWT 135512738 IC50 = 5.9 nM T36059 CI03HR 135512751 IC50 = 0.61 nM T36059 CSRL27 135512752 IC50 = 0.22 nM T36059 CV6U5T 135513694 Ki = 23 nM T36059 CTB6R7 135515408 IC50 = 1.9 nM T36059 CFQ38U 135515507 Ki = 0.5 nM T36059 C9J5WF 135516512 IC50 = 1.1 nM T36059 CCHU96 135516528 Ki = 147 nM T36059 C9C6PF 135516677 Ki = 40 nM T36059 C46YPU 135519330 Ki = 157 nM T36059 CG64XS 135522362 Ki > 1000 nM T36059 C1E2ZK 135522363 Ki > 1000 nM T36059 C2CL8J 135522364 Ki > 1000 nM T36059 C2AHQ6 135522367 Ki > 1000 nM T36059 CF9XI7 135522375 Ki > 1000 nM T36059 C4NG7Y 135522388 Ki > 1000 nM T36059 C9A7QL 135522390 Ki > 1000 nM T36059 CUNG36 135522391 Ki > 1000 nM T36059 CFJ8P2 135525108 IC50 = 5 nM T36059 C2WJI6 135529341 Ki > 1000 nM T36059 C7ARF8 135529362 Ki > 1000 nM T36059 C2V3CX 135529371 Ki > 1000 nM T36059 CVXF23 135529372 Ki > 1000 nM T36059 CJ86ZY 135529373 Ki > 1000 nM T36059 CESZ83 135529396 Ki > 1000 nM T36059 CJ4Y1H 135529398 Ki > 1000 nM T36059 C2ET0M 135533291 Ki = 39 nM T36059 C3V0NZ 135537639 IC50 = 0.23 nM T36059 C1OS2X 135542443 IC50 = 0.29 nM T36059 C8I2FM 135542466 Ki = 113 nM T36059 CR8GQ5 135542518 IC50 = 3.3 nM T36059 CU3F1O 135542558 Ki = 81 nM T36059 C51PIY 135543600 IC50 = 0.21 nM T36059 CF3UQ4 135543624 Ki = 538 nM T36059 CKN9Y0 135543763 Ki = 110 nM T36059 C6WLJ3 135544018 IC50 = 5.4 nM T36059 C1K5QE 135544028 IC50 = 0.9 nM T36059 CMOB21 135544044 IC50 = 15 nM T36059 CR6X3F 135544059 IC50 = 8.7 nM T36059 C38LZC 135545353 Ki = 220 nM T36059 CI3LK7 135546224 Ki = 600 nM T36059 C5Y9WX 135546648 Ki > 1000 nM T36059 CESD69 135546649 Ki > 1000 nM T36059 CUI90X 135546657 Ki > 1000 nM T36059 C5KX8N 135546658 Ki > 1000 nM T36059 CLX7A1 135554424 Ki = 260 nM T36059 C7KW6I 135678052 Ki > 1000 nM T36059 CLV18T 135738630 IC50 = 42 nM T36059 C26YKB 135738631 IC50 < 10 nM T36059 C27QXV 135738634 IC50 = 12 nM T36059 C1BX3M 135738635 IC50 = 130 nM T36059 C7EI9N 135738639 IC50 = 19 nM T36059 CHFQ46 135738640 IC50 < 10 nM T36059 CC4D8I 135738642 IC50 = 150 nM T36059 CE6LS4 135738644 IC50 < 10 nM T36059 C6GI3C 135738646 IC50 = 6.2 nM T36059 C67BTG 135738649 IC50 = 4.1 nM T36059 C8S9QY 135738652 IC50 = 450 nM T36059 CP17UV 135738655 IC50 < 10 nM T36059 CVKG20 135738656 IC50 = 10 nM T36059 CD6GS7 135738659 IC50 = 2.1 nM T36059 CB0N6W 135741974 Ki = 100 nM T36059 C62PTQ 135874413 Ki > 1000 nM T36059 C87ZQJ 135874414 Ki > 1000 nM T36059 C9X1UL 135874415 Ki > 1000 nM T36059 CT40VW 135874416 Ki > 1000 nM T36059 C1V9TY 135874420 Ki > 1000 nM T36059 C1T4GB 135874421 Ki > 1000 nM T36059 CFSX68 135874422 Ki > 1000 nM T36059 CNLH54 135874423 Ki > 1000 nM T36059 C2FK6J 135874424 Ki > 1000 nM T36059 C04YTD 135874425 Ki > 1000 nM T36059 CIQ04D 135874427 Ki > 1000 nM T36059 C6TO4A 135874428 Ki > 1000 nM T36059 CO0C5V 135874429 Ki > 1000 nM T36059 C9JQ2C 135874430 Ki > 1000 nM T36059 CSOV01 135874431 Ki > 1000 nM T36059 C75TGS 135874432 Ki > 1000 nM T36059 C93GBH 135874433 Ki > 1000 nM T36059 CV7US0 135874434 Ki > 1000 nM T36059 CUC4F8 135911552 Ki = 16 nM T36059 CS6PJ9 135911553 Ki = 52 nM T36059 CYX49P 135911555 Ki = 900 nM T36059 CR5I1V 135911556 Ki = 54 nM T36059 CC82BI 135911557 Ki = 1.2 nM T36059 CZ43UC 135911558 Ki = 14 nM T36059 C1D9AL 135911560 Ki = 250 nM T36059 C4FBX6 135911561 Ki = 10 nM T36059 CJ32BU 135911562 Ki = 72 nM T36059 CRM7K5 135921140 Ki = 47 nM T36059 C3R4VH 135968990 Ki = 321 nM T36059 C7JI8O 135976345 Ki = 59 nM T36059 C0NFP8 135976347 Ki = 577 nM T36059 CN2K9S 135996021 Ki = 30000 nM T36059 C0I4DH 135996022 Ki = 20500 nM T36059 CS72MI 135996023 Ki = 28800 nM T36059 C52RUZ 135996024 Ki = 21600 nM T36059 C5B6DW 135996025 Ki = 11000 nM T36059 CSAV81 136000583 Ki = 640 nM T36059 C5J1KX 136000584 Ki = 9.8 nM T36059 C7R9LG 136002185 Ki > 1000 nM T36059 C3BV1J 136002186 Ki > 1000 nM T36059 CSBL59 136002187 Ki > 1000 nM T36059 CGS18F 136002248 Ki > 1000 nM T36059 CUK9J5 136019511 Ki = 1.46 nM T36059 C09XTP 136023344 Ki = 315 nM T36059 CBZ1I4 136025838 Ki = 5.04 nM T36059 CCS5F0 136025881 Ki = 1.93 nM T36059 C2VZR6 136025990 Ki = 2.36 nM T36059 CA17MI 136026025 Ki = 24.7 nM T36059 C9SR2V 136026026 Ki = 12.2 nM T36059 C6KNF2 136026027 Ki = 3.58 nM T36059 CO90BT 136026133 Ki = 2.37 nM T36059 CM3YH2 136026181 Ki = 15 nM T36059 CT6QN3 136029178 Ki = 432 nM T36059 CGW89B 136035286 Ki = 450 nM T36059 C5VDA8 136035287 Ki = 440 nM T36059 C38LUX 136036809 Ki > 1000 nM T36059 CEHF18 136042327 Ki > 1000 nM T36059 C4U7ZM 136042328 Ki > 1000 nM T36059 CSR0Z3 136042329 Ki > 1000 nM T36059 C9C2SF 136042330 Ki > 1000 nM T36059 C75CXE 136042331 Ki > 1000 nM T36059 CS49WL 136042332 Ki > 1000 nM T36059 CQ2ZA9 136042333 Ki > 1000 nM T36059 CON2J4 136042334 Ki > 1000 nM T36059 C5VY2Z 136042335 Ki > 1000 nM T36059 CTEB06 136042336 Ki > 1000 nM T36059 CJW64L 136042337 Ki > 1000 nM T36059 C05QUF 136042338 Ki > 1000 nM T36059 C0SX1K 136042339 Ki > 1000 nM T36059 CQ37GX 136042340 Ki > 1000 nM T36059 CF3BR5 136042341 Ki > 1000 nM T36059 C75XRI 136042342 Ki > 1000 nM T36059 CS7HM2 136042343 Ki > 1000 nM T36059 C3S1WY 136042344 Ki > 1000 nM T36059 CR5H4M 136042345 Ki > 1000 nM T36059 C29YZE 136042346 Ki > 1000 nM T36059 CAP1C6 136042347 Ki > 1000 nM T36059 C5EX7D 136042348 Ki > 1000 nM T36059 C4L7GE 136042349 Ki > 1000 nM T36059 C9JM7Y 136042350 Ki > 1000 nM T36059 CO15GM 136042351 Ki > 1000 nM T36059 COEZ25 136042352 Ki > 1000 nM T36059 CGX6H7 136042353 Ki > 1000 nM T36059 C1W9XD 136042354 Ki > 1000 nM T36059 CA6TI2 136042355 Ki > 1000 nM T36059 CJ75XH 136068601 Ki = 3.85 nM T36059 CL5B7U 136068602 Ki = 21.5 nM T36059 CU6C4Z 136068688 Ki = 10.3 nM T36059 CSJE87 136068689 Ki = 13.2 nM T36059 C7SLK3 136068716 Ki = 2.38 nM T36059 CZWP52 136068717 Ki = 44.8 nM T36059 CDX2Q0 136068718 Ki = 9.2 nM T36059 CY1RT3 136068719 Ki = 2.71 nM T36059 CI1PK7 136086896 Ki = 4.56 nM T36059 C5HL7K 136086897 Ki = 6.03 nM T36059 C6VLR1 136086898 Ki = 3.01 nM T36059 CL2E0U 136086899 Ki = 17.2 nM T36059 C01GMB 136086900 Ki = 12.6 nM T36059 CA3X5T 136086901 Ki = 1.96 nM T36059 CW49CH 136086902 Ki = 3.11 nM T36059 C4F5WR 136086903 Ki = 2.52 nM T36059 CS58QU 136086904 Ki = 2.68 nM T36059 C4B1TU 136086905 Ki = 39.8 nM T36059 CMOR91 136086906 Ki = 13.9 nM T36059 C3HY9O 136086907 Ki = 12.5 nM T36059 CWF2L1 136086908 Ki = 12.2 nM T36059 CPG3E7 136226178 Ki = 101 nM T36059 CF51IY 136228031 Ki = 3930 nM T36059 C5IX2C 136236319 Ki = 5280 nM T36059 CE2F5S 137175277 Ki = 485 nM T36059 CT0WU3 137175278 Ki = 225 nM T36059 CO3SW4 137189861 Ki = 130 nM T36059 CLY6J8 137189869 Ki = 413 nM T36059 CNB27Q 137189870 Ki = 247 nM T36059 C08CWS 137189872 Ki = 868 nM T36059 CDZ07W 137631401 Ki = 1.39 nM T36059 CZ4SO1 137631450 Ki = 1.2 nM T36059 CY61SG 137631471 Ki = 0.9 nM T36059 C40FTW 137631871 Ki = 19.95 nM T36059 CE7LZ9 137632204 Ki = 3.93 nM T36059 CSM29H 137632333 Ki = 5000 nM T36059 CL5OD9 137632338 Ki = 69.4 nM T36059 CQ36UP 137632356 Ki = 50 nM T36059 CH5F6G 137632488 Ki = 996 nM T36059 C92FIL 137632746 Ki > 30000 nM T36059 CFWO04 137632925 Ki = 134 nM T36059 CJ67UL 137633007 Ki = 650 nM T36059 C3WKU1 137633041 Ki = 2.8 nM T36059 C2AG4Y 137633276 Ki = 1.96 nM T36059 CX0MK3 137633287 Ki = 2.512 nM T36059 C9SYC5 137633560 Ki = 3.56 nM T36059 CZ2HV1 137633654 Ki = 1451 nM T36059 CZC9A2 137633810 Ki = 255 nM T36059 C9YB3R 137634085 Ki = 500 nM T36059 C71MVS 137634444 EC50 > 1000 nM T36059 C97MTE 137634467 Ki = 1.2 nM T36059 C80BAO 137635053 Ki = 0.38 nM T36059 CRGN40 137635666 Ki = 392 nM T36059 CE8IS5 137636020 Ki = 7.943 nM T36059 CYL3X8 137636099 Ki = 0.345 nM T36059 CE0OA3 137636269 Ki = 10 nM T36059 C01OZS 137636323 Ki = 1054 nM T36059 CS1EO0 137636334 Ki = 67 nM T36059 CU9G8K 137636427 Ki = 21600 nM T36059 C9TUY7 137636552 Ki = 1.49 nM T36059 C6ABK1 137636769 Ki = 3.75 nM T36059 C5P9LI 137637451 Ki = 5640 nM T36059 C53RQW 137637667 Ki > 30000 nM T36059 C6Q9JG 137637685 Ki = 668 nM T36059 CCTH80 137638080 Ki = 0.386 nM T36059 CW4S1V 137638211 Ki > 30000 nM T36059 CQ8ZL2 137638623 Ki = 429 nM T36059 C3IPH7 137638940 Ki = 4.9 nM T36059 CZ9QX0 137639459 Ki = 5200 nM T36059 CTQ67J 137639588 EC50 = 281.84 nM T36059 CCG16X 137639736 Ki = 1 nM T36059 C0SC7L 137640093 Ki > 30000 nM T36059 CZ9X1O 137640416 Ki = 7360 nM T36059 C45FXO 137641603 Ki = 343 nM T36059 CG0DI3 137641858 EC50 = 346.74 nM T36059 CJ24QK 137641890 Ki = 20.5 nM T36059 C52XDH 137641906 Ki > 30000 nM T36059 CFW9R5 137641990 Ki = 1.31 nM T36059 CV81KH 137642036 Ki = 0.575 nM T36059 CE4C5Y 137642150 Ki > 30000 nM T36059 CO94EX 137642153 Ki = 2.35 nM T36059 CB8L7K 137642940 Ki = 1 nM T36059 C7K9ZB 137642980 Ki > 30000 nM T36059 C76XKJ 137643150 Ki > 30000 nM T36059 CJQD73 137643164 EC50 = 831.76 nM T36059 C9QBD7 137643462 Ki = 109.9 nM T36059 CI7LJ8 137644039 Ki = 0.631 nM T36059 CG46DW 137644190 Ki = 117 nM T36059 CPR72G 137644224 Ki = 63 nM T36059 C58QOM 137644249 Ki = 2.49 nM T36059 C4R0OC 137644481 Ki = 214 nM T36059 C6IM0N 137644606 Ki = 1.259 nM T36059 CI7B3F 137645065 Ki = 1000 nM T36059 CUW3S0 137645094 Ki = 7.7 nM T36059 CGLI82 137645223 Ki = 232 nM T36059 CF09IY 137645275 Ki > 30000 nM T36059 CCW5R0 137645696 Ki = 4.41 nM T36059 CDBT79 137645728 Ki = 11 nM T36059 C95UJV 137645798 Ki = 207 nM T36059 CJ20CU 137645935 Ki = 400 nM T36059 C8YN3Q 137646655 EC50 = 281.84 nM T36059 CER23T 137646828 EC50 = 1412.54 nM T36059 C65YKD 137646836 Ki = 2.512 nM T36059 C3MI9L 137646957 Ki = 1.5 nM T36059 CGL83H 137647102 Ki = 60 nM T36059 CC0UF1 137647420 Ki = 0.393 nM T36059 CTR96O 137647545 Ki = 3.162 nM T36059 CE9YN0 137647778 Ki = 3.35 nM T36059 CT91AP 137648111 Ki = 53 nM T36059 CCA7I4 137648143 Ki = 0.37 nM T36059 CMV8X5 137648440 Ki = 1.5 nM T36059 C1AIP8 137648928 Ki = 0.532 nM T36059 C62KVF 137649307 Ki = 14.9 nM T36059 CWH89G 137649841 EC50 = 407.38 nM T36059 CBU3Q6 137650137 Ki = 1.2 nM T36059 CIE03Y 137650221 Ki = 1.59 nM T36059 C9W3PX 137650461 EC50 = 446.68 nM T36059 CIM50G 137650899 Ki = 4.85 nM T36059 CXCA79 137650918 EC50 = 446.68 nM T36059 C26YKP 137651319 Ki > 30000 nM T36059 C8GI7E 137651519 Ki = 781 nM T36059 CEAU34 137651531 Ki = 562 nM T36059 C13AMI 137651532 Ki > 30000 nM T36059 C9M7QE 137651747 Ki = 0.806 nM T36059 C52VBU 137651751 Ki = 4.2 nM T36059 C6Z1HJ 137651756 Ki = 1200 nM T36059 C68XOV 137651967 Ki = 5.012 nM T36059 C9G7TP 137652167 Ki = 2.3 nM T36059 CVS93H 137652383 Ki = 139 nM T36059 C8T2HN 137652475 EC50 = 331.13 nM T36059 CC84NS 137652690 Ki = 6.31 nM T36059 C8I3PG 137653289 Ki = 116.5 nM T36059 CJ24ZP 137653290 Ki = 1558 nM T36059 CHYT41 137653409 EC50 = 64.57 nM T36059 CJ1R9K 137653588 Ki = 5450 nM T36059 C47UXN 137653600 Ki = 5.012 nM T36059 C9JI8V 137654164 Ki = 19.95 nM T36059 CR8K1T 137654309 Ki = 4180 nM T36059 C4VJ5C 137654976 Ki = 7.07 nM T36059 C3AE6C 137655247 Ki = 3.45 nM T36059 C0K1ZU 137655541 Ki = 7.9 nM T36059 CB80PM 137655920 Ki = 79.43 nM T36059 CDR09J 137656083 Ki = 35.2 nM T36059 CA24YS 137656139 Ki = 5280 nM T36059 COM9J7 137656299 Ki = 2.512 nM T36059 CSJ3F9 137656764 Ki = 1.9 nM T36059 C28GAV 137656845 EC50 > 1000 nM T36059 CJUE21 137656913 Ki = 1100 nM T36059 C8FK4D 137657159 Ki = 3.162 nM T36059 C08KJH 137657382 Ki = 636 nM T36059 CH8PL9 137657570 Ki = 2730 nM T36059 CW07LP 137657589 Ki = 1.76 nM T36059 CL16PU 137657616 Ki = 3.981 nM T36059 CNTX97 137657841 Ki = 4.67 nM T36059 CJ8BC7 137657926 Ki = 0.313 nM T36059 CQ9BR1 137658051 Ki = 4370 nM T36059 CBC31H 137658387 Ki > 30000 nM T36059 CH9A8M 137658761 Ki = 136 nM T36059 CV7UE3 137659204 Ki = 5159 nM T36059 CY67UM 137659236 Ki > 30000 nM T36059 CO6B8M 137659407 Ki = 1.99 nM T36059 C7VNS4 137659441 Ki = 1.2 nM T36059 CT23EA 137659930 Ki = 42 nM T36059 C1NZL8 137659963 Ki = 96 nM T36059 C5E3RI 137660421 Ki = 1.259 nM T36059 CIDG46 137660466 Ki = 98.5 nM T36059 C0Z3HK 137660877 Ki = 107.1 nM T36059 C3Y2IZ 137661132 Ki = 0.387 nM T36059 CFUM75 137661322 Ki = 667 nM T36059 C26LVX 137661505 EC50 = 123.03 nM T36059 C1DL4J 137661670 Ki = 5.17 nM T36059 C8JFE5 137661744 Ki = 3.162 nM T36059 C30DSB 137661769 Ki = 7.2 nM T36059 COM9G6 137661811 Ki > 30000 nM T36059 CT26DO 137662145 Ki = 229 nM T36059 C4VNX5 138393285 Ki = 31.62 nM T36059 CU3PW1 139248507 Ki = 0.6 nM T36059 CT1H6B 139248508 Ki = 580.1 nM T36059 CUIN96 139248509 Ki = 195.1 nM T36059 CMO14R 139248510 Ki = 1.7 nM T36059 CYN71U 139248511 Ki = 737.5 nM T36059 C5Q9PS 139248512 Ki = 1390 nM T36059 CH6PX2 139248513 Ki = 0.5 nM T36059 C93EDJ 139248514 IC50 = 428.2 nM T36059 CF4U9V 139248515 IC50 = 152.9 nM T36059 CW74BD 141536950 Ki = 9160 nM T36059 CN2LX1 144852560 Ki = 17.4 nM T36059 CBV2L5 145436760 Ki = 6.43 nM T36059 CK15TH 145436761 Ki = 157 nM T36059 C6KOB8 145436762 Ki = 23 nM T36059 CM7J2Q 145436763 Ki = 174 nM T36059 CSQL37 145436764 Ki = 3.14 nM T36059 CNP52A 145436765 Ki = 65 nM T36059 C6OFP7 145436766 Ki = 59 nM T36059 CSQ8U5 145436767 Ki = 18.2 nM T36059 C4PZ5S 145436769 Ki = 4.72 nM T36059 CI75YJ 145949481 Ki = 15.3 nM T36059 C2GVM4 145954098 Ki = 38 nM T36059 CQ9G0K 145954398 Ki = 141 nM T36059 C3RU6S 145954471 Ki = 160 nM T36059 CZX79R 145954995 Ki = 25700 nM T36059 CC0OX1 145958464 Ki = 275 nM T36059 CH7G6S 145960536 Ki = 1912 nM T36059 C9PT5Q 145960667 Ki = 548 nM T36059 C3BY8E 145960746 Ki = 749 nM T36059 CWSM81 145960813 Ki = 112 nM T36059 C5D6AI 145960873 Ki = 2274 nM T36059 C62JCL 145960933 Ki > 10000 nM T36059 CQN69Z 145961145 Ki = 2928 nM T36059 CRBY29 145961339 Ki = 446 nM T36059 C0WBV6 145961509 Ki = 2590 nM T36059 C02OQR 145961748 Ki = 725 nM T36059 C1O0GQ 145961937 Ki = 165 nM T36059 CCB0Y2 145961997 Ki = 667 nM T36059 CT8UO0 145962202 Ki > 10000 nM T36059 C3M7ZN 145962234 Ki = 3529 nM T36059 CVA89T 145962310 Ki = 1612 nM T36059 CD6X5O 145962355 Ki = 692 nM T36059 C86APL 145962364 Ki = 780 nM T36059 CH5DS7 145962529 Ki = 1519 nM T36059 C4NXC1 145962657 Ki > 10000 nM T36059 C9UYI6 145963230 Ki = 275 nM T36059 C5MD4S 145963661 Ki = 782 nM T36059 C9E0UX 145964230 Ki = 2990 nM T36059 CS0O1Z 145964662 Ki = 266 nM T36059 C01PVB 145965471 Ki = 85 nM T36059 C1ER6I 145967791 Ki = 4550 nM T36059 CY20LR 145970075 Ki = 1410 nM T36059 CP10LJ 145971798 Ki = 904 nM T36059 C8J7FL 145971923 Ki = 827 nM T36059 CZJA45 145972655 Ki = 430 nM T36059 CE23KG 145973077 Ki = 474 nM T36059 CBT7E9 145973326 Ki >= 10000 nM T36059 CB96ZI 145975418 Ki = 719 nM T36059 CZI4H3 145976828 Ki > 10000 nM T36059 CI2HN1 145977111 Ki > 10000 nM T36059 CM1R0J 145977114 Ki = 834 nM T36059 CA1YE3 145979018 Ki > 1000 nM T36059 C9VTO3 145979285 Ki = 868 nM T36059 C8DW3E 145979590 Ki > 1000 nM T36059 C5SZN2 145979632 Ki = 89 nM T36059 C43NUZ 145980000 Ki = 656 nM T36059 C9T3DG 145980225 Ki > 1000 nM T36059 COK2V5 145980546 Ki = 7.23 nM T36059 CO3Y8B 145980553 Ki = 487 nM T36059 CP92RY 145980571 Ki = 305 nM T36059 CBCH87 145980626 Ki > 1000 nM T36059 C7NJH2 145980712 Ki = 5.62 nM T36059 CHU27O 145980918 Ki > 1000 nM T36059 CMFW02 145980971 Ki = 6.73 nM T36059 CDM63O 145981315 Ki = 30.6 nM T36059 C0T4WK 145981370 Ki = 155 nM T36059 CHQ73C 145981492 Ki = 15.1 nM T36059 CA9R1X 145981583 Ki = 3.73 nM T36059 CK14YF 145981625 Ki > 1000 nM T36059 CB1Y4K 145981689 Ki > 1000 nM T36059 CX02DQ 145981864 Ki = 3.72 nM T36059 CNTY13 145982075 Ki = 7.42 nM T36059 CAI53J 145982270 Ki = 14.3 nM T36059 CHSJ14 145982423 Ki = 2000 nM T36059 C8RT4W 145982945 Ki = 107 nM T36059 C9CG6I 145984161 Ki = 17800 nM T36059 CUM74P 145984609 Ki = 646 nM T36059 C9VDN3 145985635 Ki = 1600 nM T36059 CHS8P7 145986422 Ki = 509 nM T36059 C19BNU 145986670 Ki = 190 nM T36059 CS7D6N 145986838 Ki > 1000 nM T36059 C23OKD 145986973 Ki = 572 nM T36059 CQ9AK0 145987082 Ki = 1.99 nM T36059 CJ70FS 145987226 Ki = 2.75 nM T36059 C78MWI 145987354 Ki = 248 nM T36059 C05IZF 145987813 Ki > 30000 nM T36059 CGV37C 145987819 Ki = 3.19 nM T36059 CYB95S 145987987 Ki > 1000 nM T36059 C0AF1D 145988094 Ki = 3.37 nM T36059 CD01TO 145988590 Ki = 2070 nM T36059 C3O1MT 145988709 Ki = 2660 nM T36059 CMD74V 145988733 Ki = 16.4 nM T36059 CV53QZ 145988884 Ki = 2170 nM T36059 CV6CA4 145988962 Ki = 353 nM T36059 CEM2L0 145989440 Ki = 69.9 nM T36059 CP3G4S 145989441 Ki > 1000 nM T36059 CVS17Y 145989611 Ki = 15.3 nM T36059 CB9GL1 145989764 Ki = 4920 nM T36059 CB6U5A 145989810 Ki = 602 nM T36059 C4I1EY 145990207 Ki = 521 nM T36059 CZP5T3 145990301 Ki = 108 nM T36059 CJ0A5L 145990511 Ki = 871 nM T36059 CHV8C9 145990554 Ki = 6.52 nM T36059 C3H2ZP 145990725 Ki = 6.05 nM T36059 CJ30YT 145990769 Ki = 12.5 nM T36059 C2Y8PA 145990926 Ki = 802 nM T36059 CV5XO6 145991048 Ki = 102 nM T36059 C6ZYL7 145991283 Ki = 339 nM T36059 C9YO2T 145991303 Ki = 159 nM T36059 CN7A1X 145991427 Ki = 574 nM T36059 C26OBR 145991489 Ki = 458 nM T36059 CUP48Y 145991545 Ki = 10.8 nM T36059 C8QT3X 145991607 Ki = 4320 nM T36059 C7K5ZQ 145991651 Ki = 7750 nM T36059 C8SI9A 145991749 Ki = 7.21 nM T36059 C2CB3J 145991827 Ki = 10 nM T36059 CGH8T9 145992005 Ki > 1000 nM T36059 C3QHT6 145992189 Ki = 4.88 nM T36059 CLS8P3 145992357 Ki > 1000 nM T36059 C0NUC8 145992378 Ki > 1000 nM T36059 C1MU4D 145992652 Ki = 5.02 nM T36059 CB85AS 145992677 Ki = 326 nM T36059 C94OJE 145992790 Ki = 5.21 nM T36059 C7B3FY 145992928 Ki = 6.82 nM T36059 C47DOA 145993092 Ki = 28600 nM T36059 C9KE3Y 145993107 Ki = 204 nM T36059 CW7AK5 145993147 Ki > 1000 nM T36059 CQ5Y3F 145993331 Ki = 1000 nM T36059 CZOR31 145993511 Ki = 1.71 nM T36059 CQ93KE 145993540 Ki = 5990 nM T36059 CTE42N 145993653 Ki = 1090 nM T36059 CO54SG 145993861 Ki = 508 nM T36059 C6A3RN 145993941 Ki = 1.21 nM T36059 C0EY3Q 145994002 Ki > 1000 nM T36059 CO69HC 145994068 Ki = 13000 nM T36059 C72SMW 145994175 Ki = 129 nM T36059 CE07TR 145994259 Ki = 5.08 nM T36059 C5LXC4 153605593 Ki = 10600 nM T36059 CZ53NG 153605599 Ki = 13200 nM T36059 CQ0JR3 154730931 EC50 = 0.0631 nM T36059 C2CG8J 155510487 Ki = 43.2 nM T36059 C14XVK 155510489 Ki = 99 nM T36059 CD52TC 155511687 Ki = 691 nM T36059 CPMN94 155511844 Ki = 678 nM T36059 CTV8R1 155512151 Ki = 6220 nM T36059 CM5ZA9 155512438 Ki > 1000 nM T36059 CTP3K1 155512498 Ki = 55.8 nM T36059 CX96QM 155512576 Ki = 737 nM T36059 CNF8S4 155513087 Ki = 199.53 nM T36059 C1VN3I 155513402 Ki = 6.7 nM T36059 CV35ZN 155513505 Ki = 16600 nM T36059 CGS27D 155513515 Ki = 13.76 nM T36059 CU67HI 155513890 Ki = 20.6 nM T36059 CP7UX3 155513958 Ki = 10 nM T36059 CUB2C9 155514153 Ki = 582 nM T36059 C38LUS 155514209 Ki = 604 nM T36059 CKVM85 155514248 Ki > 10000 nM T36059 CR85FY 155514357 Ki = 32.1 nM T36059 CQ7GR6 155514463 Ki = 2.8 nM T36059 CRF2B1 155514696 Ki = 948 nM T36059 CN8E1J 155514860 Ki > 1000 nM T36059 CP6C5S 155514957 Ki > 1000 nM T36059 CLJ7Y3 155515226 Ki = 2914 nM T36059 C3Z1AL 155515319 Ki = 6.51 nM T36059 C9NJT8 155515787 Ki = 251.19 nM T36059 CSJ63V 155516000 Ki = 199.53 nM T36059 CNV02U 155516016 Ki > 10000 nM T36059 CT18NO 155516071 Ki = 509 nM T36059 CLX4D7 155516277 Ki > 1000 nM T36059 CO9PI2 155516509 Ki > 10000 nM T36059 CLN52S 155516663 Ki = 100 nM T36059 C5QJ4R 155516939 Ki > 10000 nM T36059 CAH53U 155517120 Ki > 3000 nM T36059 CR59VH 155517789 Ki = 3.7 nM T36059 C0CR9Q 155518147 Ki > 1000 nM T36059 CR5VO9 155518410 Ki = 100 nM T36059 C3SAR7 155519016 Ki > 10000 nM T36059 CP74IJ 155519148 Ki = 118 nM T36059 C0EAY4 155519375 Ki = 780 nM T36059 CX1MO3 155519551 Ki = 134 nM T36059 C9HK4E 155519617 Ki = 1376 nM T36059 C5YDE2 155519621 Ki = 32 nM T36059 CEY82J 155519727 Ki = 1350 nM T36059 C5NTJ8 155519776 Ki = 190 nM T36059 C72OJY 155519986 Ki = 4097 nM T36059 C8N1CQ 155520115 Ki > 30000 nM T36059 C9PYN7 155520412 Ki = 80.5 nM T36059 CZ1S5N 155520662 Ki = 24.9 nM T36059 CY25CV 155520663 Ki > 3000 nM T36059 C7R8UB 155520744 Ki > 10000 nM T36059 CRBE64 155520811 Ki > 10000 nM T36059 CPL4Q7 155520955 Ki = 5575 nM T36059 CXW82M 155520967 Ki > 10000 nM T36059 C6A4UH 155521103 Ki = 247 nM T36059 CAC2H5 155521304 Ki > 3000 nM T36059 CS2GJ8 155521355 Ki = 48 nM T36059 C25KBM 155521478 Ki > 30000 nM T36059 CYW7Q0 155521543 Ki > 1000 nM T36059 CXD9G0 155521637 Ki = 39.81 nM T36059 CW29KY 155521694 Ki > 30000 nM T36059 C2V8SU 155521773 Ki > 10000 nM T36059 CHTX98 155522541 Ki > 1000 nM T36059 CGJ0W4 155522875 Ki > 30000 nM T36059 CBW5G4 155522899 Ki = 4.66 nM T36059 C0S4EM 155522991 Ki = 16.3 nM T36059 C3SJ9B 155523748 Ki = 2656 nM T36059 CK8RS0 155523968 Ki > 1000 nM T36059 C4ZIH2 155524032 Ki > 1000 nM T36059 CD24BF 155524446 Ki > 10000 nM T36059 C8E3HR 155524516 Ki > 1000 nM T36059 C3A9RO 155524965 Ki = 9.03 nM T36059 CYSK39 155525038 Ki = 32 nM T36059 CZX2N4 155525050 Ki > 1000 nM T36059 C1WZX5 155525062 Ki > 10000 nM T36059 C7MV3G 155525229 Ki = 9.1 nM T36059 CN1C6R 155525265 Ki = 11130 nM T36059 C8QIF6 155525396 Ki = 39.81 nM T36059 C78DHT 155525494 Ki = 8.6 nM T36059 CR6A7N 155525747 Ki = 4.9 nM T36059 CY0W2Z 155525787 Ki > 10000 nM T36059 CMG21X 155526077 Ki = 398.11 nM T36059 CBAK91 155527112 Ki = 4205 nM T36059 C5CO8R 155527265 Ki = 12.8 nM T36059 CQ1UZ5 155527318 Ki = 45.6 nM T36059 CS9U0T 155527740 Ki = 100 nM T36059 C86KIL 155527931 Ki > 10000 nM T36059 C3BEX2 155527968 Ki = 39.81 nM T36059 CL4RC9 155528080 Ki >= 10000 nM T36059 C3KA0S 155528136 Ki = 53.5 nM T36059 CR5E7W 155528403 Ki > 10000 nM T36059 C4OL2X 155528461 Ki > 10000 nM T36059 CAR75Z 155528717 Ki > 1000 nM T36059 CZ53GQ 155528757 Ki = 553 nM T36059 CXM9W5 155529088 Ki = 501.19 nM T36059 CGX6S4 155529530 Ki > 10000 nM T36059 CZ9YC8 155529872 Ki > 1000 nM T36059 C7WDL3 155530036 Ki > 10000 nM T36059 CVE30Z 155530257 Ki > 1000 nM T36059 CS2BT0 155530292 Ki = 59 nM T36059 C34VYA 155530298 Ki > 10000 nM T36059 CQT8O2 155530381 Ki > 1000 nM T36059 C3ZH9L 155530416 Ki = 19.95 nM T36059 C78JZY 155530514 Ki > 1000 nM T36059 CY3QH2 155530781 Ki > 10000 nM T36059 CN87UW 155530961 Ki = 300 nM T36059 C2YDZ8 155531112 Ki > 10000 nM T36059 C5X1QC 155531135 Ki = 15000 nM T36059 C13NXZ 155531338 Ki > 10000 nM T36059 CNVU03 155531548 Ki = 35.6 nM T36059 C3XQ9S 155531570 Ki = 2131 nM T36059 C4A3DX 155531727 Ki > 1000 nM T36059 C14GCE 155531842 Ki = 5.42 nM T36059 CQI01K 155531990 Ki > 1000 nM T36059 C7A9BH 155532173 Ki = 15 nM T36059 C21MLU 155532274 Ki > 1000 nM T36059 CXMC14 155532373 Ki > 3000 nM T36059 CVI21H 155532514 Ki > 1000 nM T36059 C86SCT 155532773 Ki > 30000 nM T36059 CQ96YB 155532918 Ki = 856 nM T36059 C9EU2D 155533104 Ki = 23400 nM T36059 CY0H3U 155533272 Ki = 37.1 nM T36059 C7R0NM 155533275 Ki = 31.62 nM T36059 CY8O6B 155533349 Ki = 2246 nM T36059 C9TLW2 155533451 Ki = 501.19 nM T36059 C8FCH7 155533611 Ki > 10000 nM T36059 C7E5OP 155533880 Ki = 2662 nM T36059 C9WO1Z 155533882 Ki > 10000 nM T36059 CH54UR 155534188 Ki = 264 nM T36059 CKM60Q 155534231 Ki > 10000 nM T36059 CW8FN0 155534473 Ki = 1199 nM T36059 C9QV4W 155534659 Ki = 61.5 nM T36059 C0R3PA 155534717 Ki > 10000 nM T36059 C4NU8B 155534836 Ki > 1000 nM T36059 CJB82P 155535066 Ki = 609 nM T36059 COT9U8 155535203 Ki = 822 nM T36059 CIH0T5 155535400 Ki > 10000 nM T36059 C67VZK 155535458 Ki = 7060 nM T36059 CI40DC 155535506 Ki > 10000 nM T36059 C38WUG 155536405 Ki = 211 nM T36059 CH6E1O 155536745 Ki > 1000 nM T36059 C6Q1EM 155536934 Ki = 2400 nM T36059 CMG75B 155537001 Ki > 10000 nM T36059 C8ZG7F 155537023 Ki = 30900 nM T36059 CWC87Q 155537599 Ki = 8.17 nM T36059 C3P8VK 155537874 Ki = 7090 nM T36059 CW75BA 155538492 Ki = 9.52 nM T36059 CD9KW3 155539920 Ki > 10000 nM T36059 CT7A3I 155540193 Ki > 10000 nM T36059 C8BHN2 155540525 Ki = 214 nM T36059 CF6ZE5 155540615 Ki > 10000 nM T36059 CK52SC 155540779 Ki = 3.24 nM T36059 C3P1ZT 155540839 Ki > 1000 nM T36059 CJ4PS8 155540888 Ki > 10000 nM T36059 C2L9TS 155540948 Ki > 1000 nM T36059 CBE65T 155541185 Ki > 10000 nM T36059 C19HQM 155541262 Ki > 1000 nM T36059 CV29BX 155541356 Ki = 79.43 nM T36059 C42QAK 155541530 Ki = 145 nM T36059 C2HX6J 155541790 Ki = 38 nM T36059 C1LU5B 155541865 Ki = 42.2 nM T36059 C9H5VC 155541975 Ki = 634000 nM T36059 C86KPX 155542492 Ki = 47.1 nM T36059 CMEW36 155542520 Ki = 668 nM T36059 CGY1J4 155542588 Ki = 174 nM T36059 CCV87Q 155542600 Ki > 1000 nM T36059 C8JY0G 155542643 Ki > 1000 nM T36059 C0BFX9 155542720 Ki > 1000 nM T36059 C06OKY 155542884 Ki = 8.2 nM T36059 C3XDT7 155543719 Ki = 84 nM T36059 CMT60C 155543832 Ki = 3820 nM T36059 C2DNQ0 155543871 Ki = 9820 nM T36059 C1QAZ9 155544096 Ki = 129 nM T36059 C89KIV 155544173 Ki = 6820 nM T36059 CR0EV6 155544177 Ki = 258 nM T36059 CH1G4C 155544368 Ki > 10000 nM T36059 C30NOS 155544777 Ki > 1000 nM T36059 CQ9Z2P 155545386 Ki = 15.73 nM T36059 CJS87Q 155545399 Ki = 116 nM T36059 C5Y4BH 155545414 Ki > 1000 nM T36059 C5HU6A 155545585 Ki > 1000 nM T36059 C45CUJ 155545762 Ki > 1000 nM T36059 CZ49CM 155545843 Ki = 128 nM T36059 CM5ZN0 155545870 Ki = 124 nM T36059 C2NKO5 155545904 Ki = 4 nM T36059 C3B0SI 155546100 Ki = 0.9 nM T36059 C95ICF 155546118 Ki = 173 nM T36059 C4BHE8 155546183 Ki > 1000 nM T36059 CL1T9K 155546550 Ki = 950 nM T36059 C6XP3U 155546562 Ki > 1000 nM T36059 C2QJR8 155546827 Ki = 16.4 nM T36059 C1X2GS 155546843 Ki > 10000 nM T36059 C1VHM5 155547186 Ki = 22000 nM T36059 CQE30Y 155547305 Ki = 585 nM T36059 CK1X5S 155547588 Ki > 1000 nM T36059 C42XEK 155547698 Ki > 10000 nM T36059 C8Q7JG 155547782 Ki > 1000 nM T36059 C35WAK 155548264 Ki > 1000 nM T36059 C6IL4E 155548476 Ki = 58.4 nM T36059 C39GTQ 155548778 Ki = 46.7 nM T36059 CY1XJ0 155548779 Ki = 9050 nM T36059 C4MIT2 155548780 Ki > 1000 nM T36059 C82STM 155549033 Ki = 7.943 nM T36059 C3NE6F 155549264 Ki > 1000 nM T36059 C9H6UQ 155549285 Ki = 158.49 nM T36059 CS57LN 155549377 Ki = 1611 nM T36059 CC45SE 155550088 Ki > 1000 nM T36059 CY7Q9N 155550159 Ki > 1000 nM T36059 C2IU1J 155550532 Ki > 1000 nM T36059 C6J5EX 155550807 Ki = 7490 nM T36059 CN2I3H 155550832 Ki = 8646 nM T36059 C4LN3W 155551750 Ki > 1000 nM T36059 CI41QF 155552117 Ki = 253 nM T36059 CA29GP 155552390 Ki = 3.58 nM T36059 CJ82KN 155552405 Ki > 1000 nM T36059 CM40UT 155552539 Ki > 1000 nM T36059 CF0W4K 155552683 Ki = 13 nM T36059 CIQH30 155552719 Ki > 1000 nM T36059 CX4P7S 155553385 Ki > 30000 nM T36059 CD42WK 155553510 Ki = 80.1 nM T36059 CNK6Z9 155553575 Ki > 1000 nM T36059 C1A5OR 155553697 Ki > 10000 nM T36059 CB75AP 155553750 Ki > 1000 nM T36059 CU1ZE5 155554091 Ki = 326 nM T36059 CFW01A 155554317 Ki = 524 nM T36059 CEK8A6 155555026 Ki = 31.62 nM T36059 C9J5ES 155555123 Ki = 106 nM T36059 C57MKC 155555241 Ki > 1000 nM T36059 CVDO87 155555721 Ki > 1000 nM T36059 CN38KO 155555854 Ki = 5170 nM T36059 CL3IB5 155555868 Ki = 312 nM T36059 CJ73SL 155556032 Ki > 1000 nM T36059 CDR63F 155556134 Ki = 91 nM T36059 C2VP0T 155556202 Ki > 10000 nM T36059 CYB6T5 155556258 Ki > 30000 nM T36059 CV9P2M 155556457 Ki > 10000 nM T36059 CC14ON 155556524 Ki > 1000 nM T36059 CNM4F3 155556727 Ki > 10000 nM T36059 C7M1VE 155556836 Ki = 13600 nM T36059 CGF0H2 155556884 Ki > 1000 nM T36059 C8QW7M 155556988 Ki > 10000 nM T36059 CL7S2P 155557016 Ki = 48.8 nM T36059 C9MWG2 155557128 Ki > 1000 nM T36059 CV21NW 155557226 Ki > 10000 nM T36059 C2F1JY 155557284 Ki > 30000 nM T36059 CDYO34 155557387 Ki = 456 nM T36059 CTSX95 155557611 Ki > 1000 nM T36059 CJ16GB 155557960 Ki > 1000 nM T36059 C8TO2W 155558029 Ki = 20 nM T36059 C0W7AL 155558312 Ki > 10000 nM T36059 CDMC47 155558350 Ki > 30000 nM T36059 C3A7MK 155558447 Ki > 1000 nM T36059 C8Z2TC 155558489 Ki > 10000 nM T36059 CJ3NY4 155558793 Ki = 14.2 nM T36059 CYX8T1 155558921 Ki = 1290 nM T36059 CIAE48 155558941 Ki > 30000 nM T36059 CVS4T6 155559056 Ki > 100000 nM T36059 CTI57G 155559203 Ki > 1000 nM T36059 C2B8NX 155559219 Ki = 8720 nM T36059 C5EC8U 155559408 Ki = 35.9 nM T36059 CP87XK 155559423 Ki > 1000 nM T36059 CMU6P5 155559511 Ki = 79.2 nM T36059 CQM64H 155559636 Ki = 253.7 nM T36059 C34ORN 155560261 Ki = 16600 nM T36059 C8B7CG 155560391 Ki > 1000 nM T36059 C73XYW 155560510 Ki > 1000 nM T36059 C3OP1F 155560545 Ki > 1000 nM T36059 CEXP80 155561009 Ki > 1000 nM T36059 CR5U7K 155561060 Ki = 794.33 nM T36059 C5KY7D 155561141 Ki > 1000 nM T36059 CGD7R4 155561189 Ki = 1220 nM T36059 C49XPN 155561350 Ki = 39.81 nM T36059 C1IA4X 155561597 Ki > 10000 nM T36059 CKG56Z 155562044 Ki = 84.4 nM T36059 CXUN73 155562096 Ki = 611 nM T36059 C6EN2B 155562182 Ki > 1000 nM T36059 CCOD50 155562467 Ki = 10.9 nM T36059 C1NF2M 155562789 Ki > 1000 nM T36059 CR8Y9K 155563119 Ki = 4.63 nM T36059 CM46KC 155563177 Ki > 1000 nM T36059 CQ19VC 155563189 Ki > 1000 nM T36059 CA27NL 155563199 Ki > 10000 nM T36059 C4N9GU 155563428 Ki = 1160 nM T36059 CJZO26 155563438 Ki > 100000 nM T36059 CPTM25 155563673 Ki > 1000 nM T36059 C5ZKN0 155563788 Ki > 1000 nM T36059 CD6QW7 155563833 Ki > 10000 nM T36059 CE2V5Y 155564179 Ki > 1000 nM T36059 C8TL6J 155564465 Ki > 1000 nM T36059 CHJ5Q8 155564753 Ki > 30000 nM T36059 CFNC10 155565326 Ki = 127 nM T36059 CKGC67 155565439 Ki > 10000 nM T36059 C8N3PQ 155565636 Ki > 1000 nM T36059 CYI54E 155565672 Ki > 1000 nM T36059 CI2CQ0 155565683 Ki > 1000 nM T36059 CB14WJ 155565911 Ki > 1000 nM T36059 CBI7N3 155566272 Ki = 9750 nM T36059 C6DQ1K 155566338 Ki = 288 nM T36059 C0VUO9 155566764 Ki > 1000 nM T36059 CN8RL3 155567003 Ki > 30000 nM T36059 CEK19O 155567253 Ki = 79.43 nM T36059 CPW8M5 155567457 Ki = 11.7 nM T36059 C7U5XT 155568271 Ki = 6.85 nM T36059 C5KNM6 155569051 Ki = 3784 nM T36059 CH86AJ 155569073 Ki > 1000 nM T36059 CQA3R5 155569370 Ki = 1140 nM T36059 CH83UM 155569483 Ki = 33.1 nM T36059 CP9TR0 10324985 Ki > 10000 nM T36059 C7Q9WY 11395785 Ki = 2.818 nM T36059 CG36QE 14775498 Ki = 0.3981 nM T36059 C4EBT3 16109359 EC50 = 2.692 nM T36059 CJZ23T 44333154 Ki = 23.6 nM T36059 CIU68M 44333155 Ki = 381 nM T36059 CV8BQ7 44333404 Ki = 55.8 nM T36059 C30UYD 44333842 Ki = 7.44 nM T36059 CCK07J 44333843 Ki = 28.1 nM T36059 CY9L6X 44593140 Ki = 0.2818 nM T36059 CXI01V 44593141 Ki = 1513.56 nM T36059 CA4B8E 44593142 Ki = 2.818 nM T36059 CTKI94 44593143 Ki = 1.096 nM T36059 C1XNL9 44593144 Ki = 1.622 nM T36059 CTV65H 44593164 Ki = 3890.45 nM T36059 CB5HY2 44593165 Ki = 3467.37 nM T36059 C9O5TS 44593166 Ki = 2691.53 nM T36059 CV3KE2 44593167 Ki = 17.38 nM T36059 CM9L8X 44593189 Ki = 85.11 nM T36059 C04ZSD 44593190 Ki = 416.87 nM T36059 CPW15H 44593191 Ki = 2.239 nM T36059 CWA84J 44593192 Ki = 0.6761 nM T36059 C4HSL0 44593193 Ki = 5.623 nM T36059 CXIZ74 44593214 Ki = 3981.07 nM T36059 CE3K5A 44593215 Ki = 4466.84 nM T36059 C9PH6N 44593216 Ki = 4.266 nM T36059 CTX91V 44593236 Ki = 0.8913 nM T36059 CPD5T2 44593237 Ki = 41.69 nM T36059 CY2Z6T 44593238 Ki = 2.951 nM T36059 CIGQ83 44593254 Ki = 3.631 nM T36059 C5UO8V 44593255 Ki = 18.2 nM T36059 CC0Y6M 44593256 Ki = 870.96 nM T36059 CF43BD 44593257 Ki = 1445.44 nM T36059 CO6UR2 44593258 Ki = 512.86 nM T36059 C81QHI 44593259 Ki = 309.03 nM T36059 C0KH6P 44593276 Ki = 354.81 nM T36059 C8YA9U 44593277 Ki = 436.52 nM T36059 C4NV8T 44593278 Ki = 346.74 nM T36059 C6F1JS 44593279 Ki = 2.188 nM T36059 CL3PD9 44593280 Ki = 2.512 nM T36059 CAM5F8 44593299 Ki = 630.96 nM T36059 CIY9R2 44593300 Ki = 27.54 nM T36059 CAXQ68 44593301 Ki = 29.51 nM T36059 CMQ39D 44593302 Ki = 7585.78 nM T36059 CP2MB9 44593303 Ki = 48977.88 nM T36059 C90IQB 46905977 Ki = 7.3 nM T36059 D00ASZ 16204411 Ki = 104 nM T36059 D00CJJ 12016636 Ki > 30000 nM T36059 D00CVD 252716 Ki = 0.56 nM T36059 D00GNW 16109429 Ki = 171 nM T36059 D00GQI 11313151 Ki = 267 nM T36059 D00JMT 210332 Ki = 660 nM T36059 D00JWA 46880333 Ki = 333 nM T36059 D00MFV 44572293 Ki > 100000 nM T36059 D00NFW 16109432 Ki = 8.5 nM T36059 D00YXE 11652061 Ki = 632 nM T36059 D01AAI 4046493 Ki = 4 nM T36059 D01CQU 5139184 Ki = 230 nM T36059 D01DPF 9802941 Ki = 7.9 nM T36059 D01NHH 16109434 Ki = 115 nM T36059 D01NTI 15366659 Ki = 920 nM T36059 D01PGY 10045125 Ki = 2.8 nM T36059 D01QBK 44572356 Ki = 11000 nM T36059 D01QYQ 6603931 Ki > 290 nM T36059 D01RAD 2303 Ki = 23500 nM T36059 D01VEU 44300688 Ki = 86 nM T36059 D01VXC 11278089 Ki = 531 nM T36059 D01VXP 16115754 Ki = 23 nM T36059 D01WNA 5248753 Ki = 27800 nM T36059 D01WXR 12253310 Ki = 237 nM T36059 D02CHG 248021 Ki = 32000 nM T36059 D02EAO 11243768 Ki = 51 nM T36059 D02FLH 16109427 Ki = 69 nM T36059 D02HOL 11849871 Ki >= 100000 nM T36059 D02HYT 11438116 Ki = 22.4 nM T36059 D02HZJ 11245073 Ki = 1300 nM T36059 D02JMR 16202727 Ki = 92.3 nM T36059 D02RBK 9904551 Ki >= 100000 nM T36059 D02SKN 10247549 Ki = 364 nM T36059 D02TEW 10754789 Ki = 188 nM T36059 D02VQK 668712 Ki = 670 nM T36059 D02WTN 11404772 Ki = 392 nM T36059 D02XPR 73124 Ki > 100000 nM T36059 D02ZZQ 44567454 Ki = 13300 nM T36059 D03FVK 16115753 Ki = 6 nM T36059 D03HBG 16203543 Ki = 260 nM T36059 D03JFX 7 Ki > 100000 nM T36059 D03NVE 10226014 Ki > 9000 nM T36059 D03POP 44420681 Ki = 3.8 nM T36059 D03RFA 657378 Ki = 72 nM T36059 D04DVT 126079 Ki = 3910 nM T36059 D04GFX 736736 Ki = 11500 nM T36059 D04JIR 69689 Ki > 100000 nM T36059 D04LZN 44572409 Ki = 6200 nM T36059 D04PJO 10612371 Ki = 99.3 nM T36059 D04PLH 10448986 Ki = 200 nM T36059 D04RHI 10813088 Ki = 7270 nM T36059 D04SDD 44436081 IC50 = 1.7 nM T36059 D04TTP 127993 Ki = 2050 nM T36059 D04UUT 135511822 Ki = 80 nM T36059 D04VYZ 16202842 Ki = 1920 nM T36059 D04WHE 247436 Ki >= 100000 nM T36059 D04WIA 135433795 Ki = 252 nM T36059 D04YUM 75929 Ki > 100000 nM T36059 D05CEJ 11211335 Ki = 3280 nM T36059 D05KEF 44418996 Ki = 25 nM T36059 D05NEM 10688595 Ki = 51 nM T36059 D05TMJ 10712256 Ki = 490 nM T36059 D05XGF 44186581 Ki > 1000 nM T36059 D05XKT 24749598 Ki = 50 nM T36059 D05ZUX 44207909 Ki >= 1000 nM T36059 D06ETD 9994776 Ki = 130 nM T36059 D06FNT 10247610 Ki = 17 nM T36059 D06GOE 135465785 Ki > 1000 nM T36059 D06GTI 135416058 Ki > 1000 nM T36059 D06KYP 44572292 Ki = 15000 nM T36059 D06NRZ 188323 Ki = 1720 nM T36059 D06QID 11660141 Ki = 68 nM T36059 D06RCT 16203429 Ki = 232 nM T36059 D06SGU 11774068 Ki > 9000 nM T36059 D06TXS 10563562 Ki = 1200 nM T36059 D06ZLJ 9885773 Ki = 13.4 nM T36059 D06ZWQ 4962866 Ki = 30.8 nM T36059 D07DOE 44447542 Ki = 35500 nM T36059 D07FGB 11709210 Ki = 9.3 nM T36059 D07FZA 135522368 Ki > 1000 nM T36059 D07HVJ 16203666 Ki = 2070 nM T36059 D07IPZ 11740439 Ki = 5.4 nM T36059 D07IYH 348130 Ki = 3400 nM T36059 D07PPM 135401232 Ki = 0.441 nM T36059 D07RSH 631105 Ki = 2650 nM T36059 D07VCN 10806465 Ki = 1160 nM T36059 D08AJS 135407706 Ki = 125 nM T36059 D08EBT 10981286 Ki = 1.1 nM T36059 D08EZI 11739042 Ki = 447 nM T36059 D08FOT 5311479 Ki > 10000 nM T36059 D08FSF 14969716 Ki = 16100 nM T36059 D08HBH 11359018 Ki = 167 nM T36059 D08JUQ 11652153 Ki = 9.4 nM T36059 D08JYX 11743895 Ki = 3 nM T36059 D08LZN 11450197 Ki = 134 nM T36059 D08NQA 57523213 EC50 = 0.3162 nM T36059 D08TSA 10045876 Ki = 3 nM T36059 D09HAM 10491577 Ki = 551 nM T36059 D09IRV 11523232 Ki = 200 nM T36059 D09JKT 24749707 Ki = 25.3 nM T36059 D09NEP 252696 Ki = 741 nM T36059 D09QLB 1908 Ki = 5890 nM T36059 D09RKX 135433658 Ki = 2.3 nM T36059 D09SUZ 24749831 Ki = 350 nM T36059 D09TBE 10710647 Ki = 8280 nM T36059 D09VOP 16203665 Ki = 360 nM T36059 D09VRX 11521761 Ki = 26 nM T36059 D0A0GA 11493677 Ki = 165 nM T36059 D0A0VT 44572291 Ki > 100000 nM T36059 D0A2WH 14969715 Ki = 4.61 nM T36059 D0A4MK 135489238 Ki > 1000 nM T36059 D0A5KG 16094571 Ki = 10.8 nM T36059 D0A6IO 5310960 Ki = 0.29 nM T36059 D0A6JX 452612 Ki = 33000 nM T36059 D0A9BZ 11605883 Ki > 1000 nM T36059 D0AI8F 12016633 Ki = 4200 nM T36059 D0AU7Y 135504122 Ki = 25 nM T36059 D0B0QW 10389852 Ki = 39 nM T36059 D0B0TX 44572355 Ki = 15000 nM T36059 D0B2NE 44598833 Ki = 0.4365 nM T36059 D0B3NZ 981611 Ki = 354 nM T36059 D0B3UE 12852 Ki = 13000 nM T36059 D0B8DR 10568125 Ki = 748 nM T36059 D0B8RQ 11427528 Ki = 147 nM T36059 D0B9CC 10869347 Ki = 6880 nM T36059 D0C1PS 12486289 Ki > 100000 nM T36059 D0C2UJ 8974 Ki = 19 nM T36059 D0C8FY 9953766 Ki = 108 nM T36059 D0CX7N 44572471 Ki = 3200 nM T36059 D0D4NS 11536096 Ki = 168 nM T36059 D0D9YL 11821203 Ki = 4440 nM T36059 D0DB7A 414707 Ki > 100000 nM T36059 D0E2FV 309375 Ki > 100000 nM T36059 D0E4LB 16115752 Ki = 4.1 nM T36059 D0E4UT 13789211 Ki > 100000 nM T36059 D0E5QE 25113696 Ki = 4430 nM T36059 D0E7YE 11462181 Ki = 49 nM T36059 D0E8RA 2773172 Ki >= 100000 nM T36059 D0E9QX 5312112 Ki = 68 nM T36059 D0F4EN 11470612 Ki = 212 nM T36059 D0FF6S 16038374 IC50 = 12000 nM T36059 D0G4WF 44378768 Ki = 4480 nM T36059 D0G5ZF 10318664 Ki = 2.3 nM T36059 D0G6BI 16203542 Ki = 90 nM T36059 D0G6VT 16202726 Ki = 110 nM T36059 D0GC7S 10640891 Ki = 76 nM T36059 D0GR6H 24749708 Ki = 182 nM T36059 D0H4RE 10640536 Ki = 180 nM T36059 D0H9BP 5697 Ki = 13.8 nM T36059 D0H9EY 10475082 Ki = 1150 nM T36059 D0HK5B 9798914 Ki > 10000 nM T36059 D0I1EP 117900 Ki = 1210 nM T36059 D0I1IW 16203539 Ki = 490 nM T36059 D0I2EQ 16109426 Ki = 61 nM T36059 D0I7HL 14842885 Ki = 66 nM T36059 D0I8GD 10065929 Ki = 7.66 nM T36059 D0IG5E 44582613 Ki = 417 nM T36059 D0IJ2X 10219753 Ki = 3080 nM T36059 D0J1BA 393594 Ki = 0.0314 nM T36059 D0J3TY 10588437 Ki = 5 nM T36059 D0J4EZ 135443359 Ki > 1000 nM T36059 D0J4SW 10731097 Ki = 3.2 nM T36059 D0JJ6T 10021483 Ki = 101 nM T36059 D0K0OT 1329 Ki = 200 nM T36059 D0K5WC 44567438 Ki = 17700 nM T36059 D0K6ZA 5311041 Ki = 450 nM T36059 D0K8ZW 10998551 Ki = 639 nM T36059 D0K8ZZ 448222 Ki = 0.8 nM T36059 D0KJ3H 16203431 Ki = 513 nM T36059 D0KT3L 10454501 Ki = 4.4 nM T36059 D0L0VU 135484064 Ki > 1000 nM T36059 D0L2MN 11529627 Ki = 94 nM T36059 D0L3BI 10593671 Ki = 3950 nM T36059 D0L5JL 1917 Ki = 1300 nM T36059 D0L6YI 16203540 Ki = 234 nM T36059 D0LD0X 128525 Ki = 2370 nM T36059 D0LP5V 11536936 Ki = 9.5 nM T36059 D0M3CG 93205 Ki = 8.7 nM T36059 D0MH4R 6716 Ki = 60000 nM T36059 D0N1PT 11500124 Ki = 140 nM T36059 D0N1QO 10320311 Ki = 4.3 nM T36059 D0N1QP 16109423 Ki = 180 nM T36059 D0N2DP 11484484 Ki = 340 nM T36059 D0N5IE 10590030 Ki = 5000 nM T36059 D0N8RM 242652 Ki > 100000 nM T36059 D0NF3E 11565524 Ki = 879 nM T36059 D0NJ4H 5281670 Ki = 34000 nM T36059 D0NO5E 7315331 Ki = 206 nM T36059 D0O0FP 9860294 Ki > 1000 nM T36059 D0O2AV 9843120 Ki = 33.3 nM T36059 D0O4KI 9834769 Ki = 1813 nM T36059 D0O6NS 81457 Ki > 10000 nM T36059 D0O8QS 10760609 Ki = 79 nM T36059 D0OR5V 414708 Ki > 100000 nM T36059 D0OX0V 11688103 Ki = 955 nM T36059 D0P0BV 16202841 Ki = 120 nM T36059 D0P5ZE 11771279 Ki = 47 nM T36059 D0P7CS 667741 Ki = 82 nM T36059 D0P7MU 4119262 Ki = 3400 nM T36059 D0P8MK 44572469 Ki > 100000 nM T36059 D0PU6F 11658819 Ki = 763 nM T36059 D0Q1RD 16202725 Ki = 296 nM T36059 D0Q3LM 16115477 Ki = 13 nM T36059 D0Q5HW 9801709 Ki = 5.9 nM T36059 D0Q6KO 1942 Ki > 100000 nM T36059 D0Q6WX 2690 Ki = 7.9 nM T36059 D0Q9GL 135443367 Ki > 1000 nM T36059 D0QN4U 16202728 Ki = 142 nM T36059 D0R1XY 123807 IC50 = 11.22 nM T36059 D0R4LZ 11536774 Ki = 4 nM T36059 D0R8OK 822296 Ki > 100000 nM T36059 D0RI4S 10636110 Ki = 74.5 nM T36059 D0RZ2M 11572592 Ki = 38 nM T36059 D0S0RK 10680 Ki = 16900 nM T36059 D0S4JI 20262 Ki > 100000 nM T36059 D0S5XP 44572408 Ki = 20000 nM T36059 D0S6QA 11608719 Ki > 100000 nM T36059 D0T2RY 9948320 Ki >= 1000 nM T36059 D0T3YY 59190723 IC50 = 1400 nM T36059 D0T7GG 16109430 Ki = 6.9 nM T36059 D0TC7N 9953255 Ki = 6.2 nM T36059 D0TU7I 5353365 Ki > 1000 nM T36059 D0V1TS 21604934 Ki = 370 nM T36059 D0V2NH 14969717 Ki = 7510 nM T36059 D0V7MX 247678 Ki > 100000 nM T36059 D0V7TA 135911551 Ki = 185 nM T36059 D0V8MD 1922 IC50 = 1250 nM T36059 D0W1PF 16109428 Ki = 7.3 nM T36059 D0W3MT 11565892 Ki = 17 nM T36059 D0W6FC 44572473 Ki >= 100000 nM T36059 D0W6TG 44186666 Ki > 10000 nM T36059 D0W8RB 44572357 Ki > 100000 nM T36059 D0WI4D 11617054 Ki = 35 nM T36059 D0X5PJ 135529391 Ki > 1000 nM T36059 D0XC9U 10500941 Ki = 317 nM T36059 D0Y5WQ 44185871 Ki > 10000 nM T36059 D0Y6HQ 16115478 Ki = 7.9 nM T36059 D0Y7HG 5281616 Ki = 3150 nM T36059 D0Y8EU 393595 Ki = 0.59 nM T36059 D0Y8LD 135529386 Ki > 1000 nM T36059 D0Y8SB 4355631 Ki = 13 nM T36059 D0Y9WZ 44583036 Ki = 422 nM T36059 D0YE5K 2241548 Ki = 410 nM T36059 D0YR1V 135457998 IC50 = 0.25 nM T36059 D0Z1WY 44447548 Ki = 18900 nM T36059 D0Z2CL 24749595 Ki = 550 nM T36059 D0Z2QM 23562742 Ki > 100000 nM T36059 D0Z3IZ 11334464 Ki = 1120 nM T36059 D0Z3XC 11185362 Ki = 6.88 nM T36059 D0Z7BC 44442164 Ki = 50 nM T36059 D0Z8NC 16109435 Ki = 637 nM T36059 D0Z8VU 44572295 Ki = 15000 nM T36059 D0ZF8N 11196622 Ki = 166 nM T36059 D0ZL2A 3661570 Ki = 18.9 nM T36059 D0ZW9L 11150373 Ki = 262 nM T77594 D00CSQ 5564 IC50 = 100000 nM T77594 D0ZX2G 3598 IC50 = 9100 nM T77594 C6A3UH 3037 IC50 = 100000 nM T77594 CA6YX9 6928 IC50 = 100000 nM T77594 C3PUL0 8398 IC50 = 100000 nM T77594 C0WK1V 16779 IC50 = 100000 nM T77594 CJIA59 75575 IC50 = 100000 nM T77594 CH2DQ1 122177324 IC50 = 300 nM T77594 D0H0AU 25195348 IC50 = 800 nM T00972 C26SVD 451777 IC50 = 250000 nM T00972 C5ZJQ3 488950 IC50 = 30000 nM T00972 C7GFT4 488962 IC50 > 100000 nM T00972 C8Q9JO 16134139 IC50 = 0.86 nM T00972 C7EC9G 16134140 IC50 = 0.84 nM T00972 C3A0YM 16134186 IC50 = 0.34 nM T00972 C6JQ3C 16143364 IC50 = 0.35 nM T00972 C6PG2R 46186917 IC50 = 9600 nM T00972 C9HL2I 46200686 IC50 = 9300 nM T00972 CRC8H5 53324414 IC50 = 83200 nM T00972 CG64CF 71596849 IC50 = 2.18 nM T00972 CZ7R4M 71597777 IC50 = 2.27 nM T00972 C8ML9U 122184656 IC50 = 17.74 nM T00972 C0FJ8S 122184657 IC50 = 17.7 nM T00972 CZ1R0G 122184658 IC50 > 2250 nM T00972 CF5P4J 122184659 IC50 = 58.79 nM T00972 D03QJA 11718722 IC50 = 1.71 nM T69375 D02NNV 3038525 IC50 > 200000 nM T69375 D03LWG 53235510 IC50 > 10000 nM T69375 D07EHV 44814409 IC50 > 10000 nM T69375 D0A6VD 25073775 IC50 = 120 nM T69375 D0E3TC 44259 IC50 = 1850 nM T69375 D0HY9S 73386890 IC50 = 76 nM T69375 D0K2ZF 22049997 IC50 > 200000 nM T69375 D0S6TK 11213558 EC50 = 10 nM T69375 D0X4MN 11597537 Ki = 6.2 nM T69375 D05SJB 10040667 IC50 = 59 nM T69375 D08DNZ 45102739 IC50 = 43 nM T69375 D09QKG 25104303 IC50 = 170 nM T69375 D0PG5N 25123232 IC50 = 4230 nM T69375 D0UY9Y 46869000 IC50 = 11900 nM T69375 D0W7MG 11647397 IC50 = 120 nM T69375 D0W8BL 46868926 IC50 = 5 nM T69375 D0ZU8L 57340689 IC50 = 0.5 nM T69375 D02MVG 11167112 IC50 = 76 nM T69375 D0A9KI 9863367 IC50 > 20 nM T69375 D0F8DL 176155 IC50 = 290 nM T69375 D0T3ME 156422 IC50 = 6 nM T69375 CIZN03 294348 IC50 = 10700 nM T69375 CHYR03 298930 IC50 = 7700 nM T69375 CCK16M 322479 IC50 = 700 nM T69375 C3NL7G 331326 IC50 = 21500 nM T69375 CZA07M 338287 IC50 = 2500 nM T69375 C0EB7O 381376 IC50 = 2200 nM T69375 CSN5H2 391320 IC50 = 14500 nM T69375 CX1Q2E 391323 IC50 = 7800 nM T69375 C1YNB7 447721 IC50 = 675 nM T69375 C73DGZ 656907 IC50 = 300 nM T69375 CXJ40G 667570 IC50 = 195 nM T69375 CKS84B 897877 IC50 = 14100 nM T69375 C3PBJ1 942437 IC50 > 50000 nM T69375 CRGB47 1228713 IC50 > 100000 nM T69375 C67OWG 1228882 IC50 > 100000 nM T69375 C5VE3K 2231029 IC50 = 13100 nM T69375 C72CNT 2747117 IC50 = 500 nM T69375 CZHL80 2808202 IC50 = 21400 nM T69375 C8WSF5 3659633 IC50 = 2980 nM T69375 CJWX69 3848929 IC50 > 200000 nM T69375 CR0DJ8 4078145 IC50 > 100000 nM T69375 C69GSP 4079571 IC50 = 22800 nM T69375 CDK3J0 5703619 IC50 = 5028 nM T69375 CA32PV 6540289 IC50 = 3100 nM T69375 C38UZJ 6852206 IC50 = 160 nM T69375 CX35YU 9553856 IC50 = 13500 nM T69375 C4Z2GW 9819930 IC50 = 8088 nM T69375 C9LI8O 9824695 IC50 > 200000 nM T69375 C1E2DV 9826083 IC50 = 47 nM T69375 C1W4JG 9872939 IC50 = 2 nM T69375 CJ4QV2 9885993 IC50 = 1500 nM T69375 COR3S2 9892736 IC50 = 650 nM T69375 C2Y3WG 9907612 IC50 = 25000 nM T69375 C5GE7T 9917045 IC50 = 3 nM T69375 C3V6WA 9930407 IC50 = 1080 nM T69375 CN0AJ9 9934347 IC50 = 42 nM T69375 C0V7UW 9958506 IC50 = 34 nM T69375 C6RI8P 9986150 IC50 = 16 nM T69375 CV8TY1 9996476 IC50 > 10000 nM T69375 C26QHZ 10005638 IC50 = 4660 nM T69375 C37AVM 10126288 IC50 > 200000 nM T69375 CJF68Z 10151092 IC50 > 200000 nM T69375 C69DHW 10158652 IC50 < 16000 nM T69375 C19GNQ 10193032 IC50 > 200000 nM T69375 CCD61V 10193155 IC50 > 200000 nM T69375 CRD0W6 10194381 IC50 > 200000 nM T69375 CJ4Q1N 10195333 IC50 > 200000 nM T69375 CA9IL4 10207537 IC50 = 1400 nM T69375 C4COW5 10216550 IC50 > 200000 nM T69375 CJF89L 10288541 IC50 > 200000 nM T69375 C3FL9K 10295633 IC50 > 10000 nM T69375 C7SFI1 10296883 IC50 > 10000 nM T69375 CPS9U3 10319232 IC50 > 10000 nM T69375 CIS0N3 10323382 IC50 = 1750 nM T69375 CA8B5T 10390073 IC50 = 261 nM T69375 CD47LT 10522840 IC50 = 910 nM T69375 CN2TU0 10526792 IC50 = 98 nM T69375 CA91SJ 10529636 IC50 = 735 nM T69375 CXN40D 10565927 IC50 = 130 nM T69375 CGSD37 10567785 IC50 = 29 nM T69375 CFP95Y 10591281 IC50 = 180 nM T69375 CW1L8E 10591928 IC50 = 140 nM T69375 CJ2O7T 10601190 IC50 = 295 nM T69375 CY7ER5 10620296 IC50 = 3300 nM T69375 C16KBG 10637813 IC50 = 1420 nM T69375 CLSA43 10663963 IC50 = 175 nM T69375 CKZ95C 10829684 IC50 = 210 nM T69375 CA53TB 10972838 IC50 = 1800 nM T69375 C6D9HX 11155124 IC50 > 200000 nM T69375 CK4DN6 11178413 IC50 > 200000 nM T69375 C5HRC0 11268703 IC50 > 200000 nM T69375 CEA01Q 11270757 IC50 > 200000 nM T69375 CBOP58 11293798 Ki > 10000 nM T69375 CUQK84 11305782 IC50 > 200000 nM T69375 C26BZX 11362471 Ki > 10000 nM T69375 C9N0VD 11385711 IC50 > 200000 nM T69375 C3JI9L 11396732 IC50 > 200000 nM T69375 CH7KE1 11397096 IC50 > 200000 nM T69375 CWXB93 11397177 Ki > 10000 nM T69375 C0APW4 11422034 IC50 = 220 nM T69375 CB4E7Q 11430712 IC50 > 200000 nM T69375 CTUM34 11431185 IC50 = 167000 nM T69375 C84SZX 11442171 IC50 > 200000 nM T69375 C7UVM8 11492814 IC50 > 10000 nM T69375 CH6XL5 11493316 IC50 = 740 nM T69375 CRS89T 11499625 IC50 = 470 nM T69375 CCV71Z 11500561 IC50 = 790 nM T69375 CXBU49 11502255 IC50 = 404000 nM T69375 CU0QR2 11509379 IC50 > 10000 nM T69375 CY20KH 11514465 IC50 = 3500 nM T69375 CLC92Y 11514477 IC50 > 10000 nM T69375 C7H6PZ 11516913 IC50 = 100 nM T69375 CH2IZ9 11517688 IC50 = 8300 nM T69375 CJ9OH7 11538129 IC50 = 250 nM T69375 CTG83F 11539329 IC50 = 150 nM T69375 C4U3YQ 11543503 IC50 = 4900 nM T69375 CJ97XP 11544489 IC50 = 610 nM T69375 CF7JG0 11551231 IC50 = 3400 nM T69375 CM57ZU 11553156 IC50 = 180 nM T69375 C7DX5S 11558435 IC50 = 770 nM T69375 C5VML9 11558444 IC50 > 10000 nM T69375 C4I0YH 11558900 IC50 = 310 nM T69375 C3KT8X 11559766 IC50 = 240 nM T69375 CVS32L 11560956 IC50 = 46 nM T69375 C70ROB 11564900 IC50 = 3000 nM T69375 C78ZTX 11565848 IC50 = 5100 nM T69375 CT3S1G 11568224 IC50 = 100000 nM T69375 CK9D6M 11579435 IC50 > 10000 nM T69375 C9XBP4 11580158 IC50 = 6300 nM T69375 CYK05Q 11586583 IC50 > 10000 nM T69375 C6O0HX 11587896 IC50 = 260 nM T69375 C24JGU 11589125 IC50 = 270 nM T69375 CQ82SM 11589163 IC50 = 130 nM T69375 CMIL86 11590363 IC50 = 70 nM T69375 C4S3JZ 11600899 IC50 = 4500 nM T69375 CB59ND 11601122 IC50 > 10000 nM T69375 CZ70BL 11601246 IC50 = 8400 nM T69375 CVH94J 11601374 IC50 > 10000 nM T69375 CUK87R 11602023 IC50 = 360 nM T69375 CQ29WV 11602291 IC50 = 274 nM T69375 C7TXB8 11609198 IC50 = 1200 nM T69375 C1A4SV 11615890 IC50 = 690 nM T69375 C73PTY 11616278 IC50 > 10000 nM T69375 C5B3XJ 11620410 IC50 > 40000 nM T69375 COT15X 11622644 IC50 > 10000 nM T69375 CFD43W 11624410 IC50 > 10000 nM T69375 CHB3F2 11626055 IC50 = 198 nM T69375 CSNY14 11638719 IC50 > 10000 nM T69375 C9T6SC 11640926 IC50 = 64 nM T69375 C6NO5B 11647280 IC50 = 26 nM T69375 C5ENI8 11651832 IC50 = 2900 nM T69375 C9VP4Y 11655237 IC50 = 49 nM T69375 CX1T5L 11666890 IC50 = 640 nM T69375 CKDU79 11666971 IC50 > 10000 nM T69375 C4CF9O 11667089 IC50 = 900 nM T69375 CV6Y3Z 11673227 IC50 > 10000 nM T69375 C9GN5Y 11674342 IC50 = 4900 nM T69375 CY5TR4 11680140 IC50 > 10000 nM T69375 CJ9KN7 11683817 IC50 > 10000 nM T69375 C2CPZ3 11695458 IC50 = 740 nM T69375 C9I7QG 11697773 IC50 = 740 nM T69375 C0SU9F 11697791 IC50 > 100000 nM T69375 CM1KG9 11705144 IC50 > 10000 nM T69375 CVC2S4 11722798 IC50 > 10000 nM T69375 CBC08P 11846124 IC50 = 120 nM T69375 CD60CH 11846125 IC50 = 53 nM T69375 C5LIW2 11846126 IC50 = 41 nM T69375 CNJB87 11846287 IC50 = 11 nM T69375 CEMS06 11846288 IC50 > 10000 nM T69375 CX8B0G 11846458 IC50 = 610 nM T69375 CIJ93W 11846459 IC50 = 120 nM T69375 C5KC7Q 11846461 IC50 = 190 nM T69375 CAZS08 11848309 IC50 = 5954 nM T69375 C43IVN 11848567 IC50 > 10000 nM T69375 C9LAY8 11848825 IC50 = 4831 nM T69375 CHR92S 11858109 IC50 > 100000 nM T69375 CC09DE 11955790 IC50 = 37 nM T69375 C8E4TS 11992146 IC50 = 21000 nM T69375 CXU6M2 12310041 IC50 = 2200 nM T69375 CEX45S 12723726 IC50 = 9300 nM T69375 CBF4X2 15991561 IC50 = 5011.87 nM T69375 CFPW41 16007116 IC50 = 74 nM T69375 C9TU1O 16046126 IC50 > 1000 nM T69375 C3V6EX 16049812 IC50 = 38 nM T69375 CKR57M 16086104 IC50 > 25000 nM T69375 C16NRY 16086114 IC50 = 173 nM T69375 CZL8G5 16115351 IC50 = 1280 nM T69375 CGC34R 16118737 IC50 = 4290 nM T69375 C5VPH9 16129448 IC50 = 433 nM T69375 C0C5AZ 16129582 IC50 = 25 nM T69375 C6L9VD 16216351 IC50 = 47 nM T69375 CU56EW 16664858 IC50 = 316.23 nM T69375 C3F8HS 16721052 IC50 = 5500 nM T69375 C7I9VO 21088983 IC50 > 200000 nM T69375 C3ZUL4 22050022 IC50 > 200000 nM T69375 CN60BZ 22050201 IC50 > 200000 nM T69375 C1M5DE 22050258 IC50 > 200000 nM T69375 CI1NV9 22050379 IC50 > 200000 nM T69375 CJ58LI 22050440 IC50 > 200000 nM T69375 C13EYW 22050442 IC50 > 200000 nM T69375 CH5FW9 22050449 IC50 > 200000 nM T69375 C09RGX 22050478 IC50 > 200000 nM T69375 CM95IS 22050722 IC50 > 171000 nM T69375 CSH4R3 22050741 IC50 > 200000 nM T69375 C9WF3I 22050830 IC50 > 200000 nM T69375 CUM74N 22051118 IC50 > 200000 nM T69375 CM2UY0 23647201 IC50 = 3000 nM T69375 CGXB32 23647237 IC50 = 68 nM T69375 CBV3A2 23647238 IC50 = 4400 nM T69375 CDMI50 23661564 IC50 > 200000 nM T69375 CVOT06 24535122 IC50 > 50000 nM T69375 CV9U8E 24745781 IC50 > 10000 nM T69375 C7YG1N 24759534 IC50 = 850 nM T69375 CQNP54 24764449 IC50 = 100000 nM T69375 C4Z9CN 24769780 IC50 = 4700 nM T69375 C16DKC 24810995 IC50 = 1000 nM T69375 CC8Y1U 24810996 IC50 = 140 nM T69375 CH21WG 24810997 IC50 = 83 nM T69375 CQ1D8M 24810999 IC50 = 430 nM T69375 CNI4W8 24811099 IC50 = 360 nM T69375 C0MXK3 24811100 IC50 = 140 nM T69375 CFZN51 24811101 IC50 = 66 nM T69375 CRF71M 24811102 IC50 = 46 nM T69375 CB8A2T 24811103 IC50 > 10000 nM T69375 CJ7M8K 24823663 IC50 = 97 nM T69375 CLP68C 24823665 IC50 = 110 nM T69375 CRV5C7 24823814 IC50 = 230 nM T69375 CSW3D9 24823964 IC50 = 180 nM T69375 CL61YV 24824104 IC50 = 170 nM T69375 CX0S9L 24854902 IC50 = 4390 nM T69375 C1SVT2 24854903 IC50 = 7772 nM T69375 C4OWF8 24875373 IC50 = 123 nM T69375 CY8L7E 24896769 IC50 > 10000 nM T69375 C8DG1Y 24941253 IC50 = 5524 nM T69375 C42HGN 24957306 IC50 = 350 nM T69375 CK4W5P 24957308 IC50 = 360 nM T69375 CE8KJ9 24960632 IC50 = 720 nM T69375 C9WOQ0 24960635 IC50 = 650 nM T69375 C6B0IM 24961360 IC50 = 178 nM T69375 CU7I2E 24963046 IC50 = 629 nM T69375 CD0TB3 25024184 IC50 = 339 nM T69375 C0JT3O 25065992 IC50 = 11 nM T69375 CB5TY4 25066206 IC50 = 75 nM T69375 CX2J3S 25066411 IC50 = 269 nM T69375 CM04RX 25066412 IC50 = 418 nM T69375 CG34VQ 25066413 IC50 = 3170 nM T69375 CJRG97 25066414 IC50 = 2700 nM T69375 CN9SJ7 25066415 IC50 = 38 nM T69375 C7IM8Q 25066416 IC50 = 649 nM T69375 C57TQU 25066617 IC50 = 1420 nM T69375 C7BI0O 25066619 IC50 = 2200 nM T69375 C6NU1D 25071599 IC50 = 1410 nM T69375 CXD9K3 25071600 IC50 = 90 nM T69375 CM2K9V 25119432 IC50 = 176 nM T69375 CF7C5B 25129829 IC50 > 10000 nM T69375 CXNM84 25129830 IC50 = 9685 nM T69375 CY2S1P 25129831 IC50 > 10000 nM T69375 CTO24B 25174101 IC50 = 70 nM T69375 CYTV68 25181985 IC50 = 28 nM T69375 C5KIE7 25182113 IC50 = 50 nM T69375 CMF51N 25222038 IC50 = 99 nM T69375 CV7AG6 25660569 IC50 = 14600 nM T69375 C5GZ8L 26704995 IC50 > 50000 nM T69375 CE0PX2 42601396 IC50 = 570 nM T69375 CGV34B 42608443 IC50 = 1400 nM T69375 CM0C2R 42608444 IC50 = 150 nM T69375 CI5AE0 43623574 IC50 > 50000 nM T69375 CX16AN 44138038 Ki = 17 nM T69375 CO42DC 44138048 IC50 = 794.33 nM T69375 CL65QV 44138049 IC50 = 1258.93 nM T69375 C75TAQ 44200209 IC50 = 50 nM T69375 C7W4AX 44200211 IC50 = 590 nM T69375 C16HSY 44200344 IC50 = 82 nM T69375 CBY7T8 44200468 IC50 > 3000 nM T69375 C0KD4U 44346053 IC50 = 30 nM T69375 CH0O5Q 44346322 IC50 > 10000 nM T69375 CY6EW5 44419110 IC50 = 300 nM T69375 CG90BS 44419115 IC50 > 10000 nM T69375 C9IWT5 44419118 IC50 = 4610 nM T69375 CNJ5F1 44419119 IC50 = 4320 nM T69375 CAYL35 44419128 IC50 = 840 nM T69375 COC4P2 44419129 IC50 = 1000 nM T69375 CH8WZ7 44419135 IC50 = 240 nM T69375 CRI6V9 44419136 IC50 = 600 nM T69375 CY6DK0 44419137 IC50 = 87 nM T69375 CZP46I 44419138 IC50 = 81 nM T69375 CQT30U 44419143 IC50 = 97 nM T69375 C8J6MZ 44419144 IC50 = 390 nM T69375 CYM3X7 44419145 IC50 = 180 nM T69375 CHG96R 44419146 IC50 = 150 nM T69375 CLX1B5 44419150 IC50 = 530 nM T69375 C0CLT1 44419151 IC50 = 160 nM T69375 CKL2A8 44419152 IC50 = 210 nM T69375 CJ1RE0 44419155 IC50 = 680 nM T69375 CQW93F 44419157 IC50 = 9200 nM T69375 CMCF90 44419158 IC50 = 30 nM T69375 C40QDE 44419161 IC50 = 340 nM T69375 C3JW9E 44419162 IC50 = 660 nM T69375 CNX3P1 44419163 IC50 = 320 nM T69375 C3GV8D 44419164 IC50 = 1400 nM T69375 C1XI7E 44419168 IC50 = 860 nM T69375 CDIL57 44419169 IC50 = 230 nM T69375 C4YQD8 44419170 IC50 = 100 nM T69375 CQE6D3 44419174 IC50 = 260 nM T69375 C76JCA 44419175 IC50 = 1290 nM T69375 CK4Z6B 44419182 IC50 = 240 nM T69375 CST57V 44419183 IC50 = 430 nM T69375 CR9ON4 44419190 IC50 = 6920 nM T69375 C1RL3U 44419191 IC50 = 120 nM T69375 C8IJ2U 44419202 IC50 = 370 nM T69375 C5KBX0 44419203 IC50 = 610 nM T69375 CRGD85 44419210 IC50 = 450 nM T69375 CP1C8D 44419211 IC50 = 84 nM T69375 CO9AK1 44419214 IC50 = 1460 nM T69375 CE20PN 44419215 IC50 = 4130 nM T69375 C4V6YN 44419216 IC50 = 69 nM T69375 CF4I1R 44419217 IC50 = 160 nM T69375 C13EQD 44419220 IC50 = 4160 nM T69375 C1KQL5 44419221 IC50 = 1790 nM T69375 CD8EB4 44419222 IC50 = 290 nM T69375 CCBL15 44419223 IC50 = 4700 nM T69375 CY1Q7N 44419226 IC50 = 300 nM T69375 CXR83C 44419227 IC50 = 969 nM T69375 CAX8F5 44440161 IC50 = 67 nM T69375 CK9H1G 44440214 IC50 = 245 nM T69375 CDF70Q 44440215 IC50 = 55 nM T69375 CK8L4U 44440216 IC50 = 709 nM T69375 CM2E3N 44440217 IC50 = 281 nM T69375 CWL30H 44440218 IC50 = 512 nM T69375 C6RD3G 44440219 IC50 = 177 nM T69375 CIAJ70 44440220 IC50 = 1551 nM T69375 C52CDB 44440221 IC50 = 15 nM T69375 C2OC7L 44440222 IC50 = 267 nM T69375 CFZS24 44440223 IC50 = 88 nM T69375 CSA87R 44440224 IC50 = 31 nM T69375 CH76CV 44440225 IC50 = 22 nM T69375 CP80UK 44440226 IC50 = 37 nM T69375 CFI06W 44440227 IC50 = 26 nM T69375 CKSO82 44440228 IC50 = 85 nM T69375 C8HWI1 44440229 IC50 = 45 nM T69375 CVD97U 44440230 IC50 = 14 nM T69375 C1B0TO 44440234 IC50 = 62 nM T69375 CS5PY4 44440235 IC50 = 698 nM T69375 C9AV4C 44440236 IC50 = 5 nM T69375 CV1G4E 44462686 IC50 = 100 nM T69375 CFK1A5 44473625 IC50 = 440 nM T69375 CU80BP 44517743 IC50 > 10000 nM T69375 CF90OX 44576212 IC50 = 166000 nM T69375 CC5W9J 44586319 IC50 = 1760 nM T69375 C5Z3LI 44591740 IC50 = 17 nM T69375 CV8F0R 44593854 IC50 = 10000 nM T69375 CJ0LU4 45104966 IC50 = 1838 nM T69375 CY3HW5 46224684 IC50 = 4100 nM T69375 C6M7CK 46232266 IC50 = 470 nM T69375 CJZA45 46232267 IC50 = 290 nM T69375 C6EX9F 46232268 IC50 = 100 nM T69375 C3PLE6 46232269 IC50 = 160 nM T69375 C3U8HV 46232270 IC50 = 100 nM T69375 CYA73D 46232312 IC50 = 140 nM T69375 C9JDL8 46232313 IC50 = 10000 nM T69375 C9JE6X 46830346 IC50 > 200000 nM T69375 CW2G7D 46868853 IC50 = 26 nM T69375 CR57OZ 46868855 IC50 = 1300 nM T69375 CI8YE5 46868856 IC50 = 41 nM T69375 C94EPL 46868925 IC50 = 15 nM T69375 C0GU4D 46868930 IC50 = 270 nM T69375 C9ULP0 46869071 IC50 = 27100 nM T69375 CU52JS 46869075 IC50 > 50000 nM T69375 CFQT10 46869147 IC50 > 50000 nM T69375 CEK2I5 46869149 IC50 = 2600 nM T69375 C2XQ4K 46869223 IC50 = 1500 nM T69375 C8U1AH 46869285 IC50 = 18 nM T69375 CKTD23 46869290 IC50 = 24 nM T69375 CV57OI 46869490 IC50 = 53 nM T69375 C9XHK0 46869491 IC50 = 38 nM T69375 C47JSD 46869493 IC50 = 36 nM T69375 C65NDB 46869609 IC50 > 50000 nM T69375 CP2A4Y 46869611 IC50 = 2400 nM T69375 CQ0AU8 46869671 IC50 > 50000 nM T69375 C4RS7M 46869672 IC50 = 824 nM T69375 C1VZM6 46869673 IC50 = 9 nM T69375 CYI69K 46869674 IC50 = 42 nM T69375 C2PC6T 46869677 IC50 = 5000 nM T69375 CSL2N6 46869740 IC50 = 15000 nM T69375 C6V9CD 46869741 IC50 = 31 nM T69375 CZCQ05 46869742 IC50 = 8700 nM T69375 C09GAW 46869745 IC50 = 125 nM T69375 CVBG98 46869815 IC50 = 230 nM T69375 CU2D5N 46869816 IC50 = 42 nM T69375 C8WH7Q 46869817 IC50 = 81 nM T69375 CFOX43 46869876 IC50 = 1620 nM T69375 CE0CY1 46869877 IC50 = 710 nM T69375 C2DW6T 46869878 IC50 = 50 nM T69375 C19DQG 46869879 IC50 = 90 nM T69375 CR1OH0 46869880 IC50 = 8 nM T69375 C8SFI1 46869881 IC50 = 21 nM T69375 CD1YH9 46869882 IC50 = 42 nM T69375 CLS29B 46872626 IC50 > 10000 nM T69375 CHU3Z8 46882355 IC50 > 200000 nM T69375 CZ47SV 46882356 IC50 > 200000 nM T69375 CSH38Q 46882357 IC50 > 200000 nM T69375 C6Z0YR 46882358 IC50 > 200000 nM T69375 C5NG6O 46882404 IC50 > 200000 nM T69375 CSX7Y1 46882405 IC50 > 200000 nM T69375 CRQ5E3 46882406 IC50 > 200000 nM T69375 C1C0YG 46882407 IC50 > 200000 nM T69375 C2KMV1 46882408 IC50 > 200000 nM T69375 CZ15LR 46882469 IC50 > 200000 nM T69375 CRKV43 46884199 Ki = 6 nM T69375 C0E6XI 46887066 IC50 > 200000 nM T69375 CNQM15 46887067 IC50 > 200000 nM T69375 C7VGU9 46887068 IC50 > 200000 nM T69375 C0JQ8T 46887097 IC50 > 200000 nM T69375 C5LAW7 46887098 IC50 > 200000 nM T69375 CM6CO3 46887099 IC50 > 200000 nM T69375 CT78EQ 46887100 IC50 > 200000 nM T69375 C38LYC 46887134 IC50 > 200000 nM T69375 C6JEI1 46887135 IC50 > 200000 nM T69375 C6L1VH 46887136 IC50 > 200000 nM T69375 C2WM7V 46887184 IC50 > 200000 nM T69375 C1VZ0G 46887185 IC50 > 200000 nM T69375 C3O8AM 46887186 IC50 > 200000 nM T69375 CGX79T 46896670 IC50 = 250 nM T69375 C60GAV 46929544 IC50 > 8000 nM T69375 CP34VL 46929748 IC50 > 1000 nM T69375 CJ2E9Q 46929857 IC50 > 25000 nM T69375 CHSF07 49806372 IC50 > 1000 nM T69375 CS18HZ 49839481 IC50 = 470 nM T69375 CH4FY5 50941455 IC50 = 69 nM T69375 CBR71Y 50941538 IC50 = 97 nM T69375 C4BN7W 50941539 IC50 = 97 nM T69375 C1LD0P 50943125 IC50 = 12 nM T69375 CI0Z7D 50943202 IC50 = 27 nM T69375 CHIY40 50943203 IC50 = 17 nM T69375 CEOB58 50943512 IC50 = 180 nM T69375 CGZC83 50943588 IC50 = 24 nM T69375 CEX3H8 50943666 IC50 = 36 nM T69375 C1JY2U 50943668 IC50 = 68 nM T69375 CPS4I5 50943669 IC50 = 20 nM T69375 C83EZX 50943670 IC50 = 49 nM T69375 CNUZ80 50943753 IC50 = 66 nM T69375 COU4W2 50943754 IC50 = 33 nM T69375 C2J7ZP 50943755 IC50 = 40 nM T69375 C5GPU9 51346941 IC50 = 90 nM T69375 CA7HQ9 52941011 IC50 = 46600 nM T69375 CA6BH5 52941226 IC50 = 26700 nM T69375 CMXC68 52941286 IC50 = 5700 nM T69375 C0DSA8 52941649 IC50 > 50000 nM T69375 C3BKR7 52942436 IC50 = 23600 nM T69375 C8R9SA 52942482 IC50 > 50000 nM T69375 CAC3J5 52942507 IC50 = 7600 nM T69375 CTPH98 52942532 IC50 > 50000 nM T69375 CS8VA0 52943431 IC50 > 50000 nM T69375 CJU79I 52943626 IC50 = 9900 nM T69375 C07JYV 52944873 IC50 = 16300 nM T69375 CB1UJ7 52944909 IC50 = 5300 nM T69375 CD2WZ5 52944914 IC50 > 50000 nM T69375 CY9B7D 52944962 IC50 > 50000 nM T69375 C1Z7KR 52946059 IC50 > 50000 nM T69375 CCMX82 52946092 IC50 > 50000 nM T69375 CPIK13 52946145 IC50 = 35000 nM T69375 C67TBV 52946152 IC50 = 47700 nM T69375 C6OH8X 52946172 IC50 > 50000 nM T69375 CC6Z1J 52947386 IC50 > 50000 nM T69375 CC5P4R 52947399 IC50 > 50000 nM T69375 C9O7FN 52947421 IC50 > 50000 nM T69375 C72TPI 52947422 IC50 > 50000 nM T69375 C3R4FI 52948519 IC50 = 3000 nM T69375 CLU92X 52948565 IC50 > 50000 nM T69375 CDXL70 52948593 IC50 = 2000 nM T69375 CO3EL9 52948602 IC50 > 50000 nM T69375 C3WHA1 52949737 IC50 > 50000 nM T69375 CMT75N 52949817 IC50 = 3100 nM T69375 CBAD62 52949818 IC50 = 3000 nM T69375 CSOB70 52950113 IC50 > 50000 nM T69375 CW2KE5 53317337 IC50 > 50000 nM T69375 CJQN83 53317338 IC50 = 28400 nM T69375 CJ2P3V 53317339 IC50 = 4524 nM T69375 C9E3FV 53317340 IC50 = 2571 nM T69375 CBTX53 53317412 IC50 = 32000 nM T69375 COCN94 53317413 IC50 = 110 nM T69375 CHC29T 53317414 IC50 = 650 nM T69375 C82LCE 53317415 IC50 = 4400 nM T69375 CR0DJ1 53317416 IC50 = 320 nM T69375 C28JAP 53317417 IC50 = 170 nM T69375 C8Q0OR 53318506 IC50 = 863 nM T69375 CP7T3N 53318709 IC50 = 380 nM T69375 CKD47I 53319944 IC50 = 613 nM T69375 CP7BR1 53319945 IC50 = 4150 nM T69375 C3TAC2 53320021 IC50 > 5000 nM T69375 COPI53 53321333 IC50 = 1500 nM T69375 C0GLS5 53321334 IC50 = 440 nM T69375 C2V0QU 53321577 IC50 = 950 nM T69375 CG8KC9 53322569 IC50 = 22500 nM T69375 C3SA1K 53322570 IC50 = 930 nM T69375 COG9J2 53322644 IC50 = 350 nM T69375 CUR1A6 53322645 IC50 = 190 nM T69375 C25OEY 53322984 IC50 = 703 nM T69375 CK8Y5F 53323911 IC50 = 765 nM T69375 C9SHJ0 53323985 IC50 = 250 nM T69375 C49MDG 53323986 IC50 = 220 nM T69375 C3AVG0 53323987 IC50 = 780 nM T69375 C18SCR 53323988 IC50 = 150 nM T69375 C38RXW 53323989 IC50 = 61 nM T69375 CXWB94 53325188 IC50 = 409 nM T69375 C8VPW5 53325283 IC50 = 93 nM T69375 CA3X2Q 53325284 IC50 = 390 nM T69375 CIG7X9 53325285 IC50 = 570 nM T69375 C4A8JK 53325286 IC50 = 150 nM T69375 CI1RT4 53325287 IC50 = 2000 nM T69375 CNT50E 53325288 IC50 = 58 nM T69375 CR91NJ 53325555 IC50 = 3140 nM T69375 CBW0G7 53326484 IC50 = 6290 nM T69375 CV7I4O 53326555 IC50 = 130 nM T69375 C27IBZ 53326556 IC50 = 470 nM T69375 C5UK3J 53326557 IC50 = 5300 nM T69375 CVJ6K9 53326558 IC50 = 530 nM T69375 C8NA4L 53384644 IC50 = 9800 nM T69375 CD0ZI6 53469858 IC50 = 864 nM T69375 CEP18Y 54581359 IC50 > 50000 nM T69375 C6JPE1 54581360 IC50 = 66.5 nM T69375 CD2YU5 54581361 IC50 = 19000 nM T69375 C49RNQ 54581362 IC50 = 4880 nM T69375 CA8U3P 54581363 IC50 > 50000 nM T69375 C5V6OY 54582175 IC50 > 30000 nM T69375 CCO5I2 54583368 IC50 = 37900 nM T69375 CECO89 54583369 IC50 = 6390 nM T69375 CRKI30 54584315 IC50 = 2250 nM T69375 C3P2HM 54584316 IC50 > 50000 nM T69375 CL69AG 54584317 IC50 = 1220 nM T69375 CC8YN2 54585285 IC50 = 15300 nM T69375 CGA8X9 54585286 IC50 > 50000 nM T69375 CV69FU 54585287 IC50 > 50000 nM T69375 CR1X8Y 54585288 IC50 = 504 nM T69375 CTY84H 54585289 IC50 > 50000 nM T69375 CWE79L 54585290 IC50 = 18600 nM T69375 C0FAG2 54585291 IC50 = 9310 nM T69375 CNLU49 54585292 IC50 = 18100 nM T69375 CNUP53 54586040 IC50 = 1900 nM T69375 CUD8J0 54586233 IC50 > 50000 nM T69375 CA5N6I 54587258 IC50 = 34600 nM T69375 CKX15Q 54587259 IC50 = 46200 nM T69375 CKQS27 54587260 IC50 = 34000 nM T69375 C57LBW 54587261 IC50 = 9140 nM T69375 C1XS2J 54760383 IC50 = 1500 nM T69375 CM8JX1 56604907 IC50 = 100000 nM T69375 CG78UW 56658171 IC50 = 62 nM T69375 C7LDZ3 56658303 IC50 = 337 nM T69375 C0MW6D 56658304 IC50 = 74 nM T69375 CS68PK 56659526 IC50 > 200000 nM T69375 CK18JP 56661802 IC50 = 140 nM T69375 CE1O3B 56661803 IC50 = 32 nM T69375 CSJ6A9 56665092 IC50 = 13 nM T69375 C7HA6J 56665093 IC50 = 17 nM T69375 CS5HP6 56665245 IC50 = 92 nM T69375 C4SO3M 56665246 IC50 = 21 nM T69375 CE2PY0 56665247 IC50 = 12 nM T69375 C9AW1E 56668539 IC50 = 145 nM T69375 C0MR6D 56668696 IC50 = 8 nM T69375 CXF3R9 56668697 IC50 = 68 nM T69375 C02JLF 56669835 IC50 = 547 nM T69375 CU3I2J 56672173 IC50 = 193 nM T69375 CJ9I6K 56672174 IC50 = 10 nM T69375 CD5NZ4 56672175 IC50 = 66 nM T69375 CRAK61 56675421 IC50 = 29 nM T69375 C3RDY2 56676664 IC50 = 1 nM T69375 C5GZ1O 56676665 IC50 = 30 nM T69375 CG3ZU0 56678888 IC50 = 164 nM T69375 CAP1M2 56682209 IC50 = 68 nM T69375 C9DO8G 56682210 IC50 = 10 nM T69375 CTO6N5 56834943 IC50 = 25 nM T69375 C97SLT 57340680 IC50 = 1140 nM T69375 C0UDN5 57340685 IC50 = 0.7 nM T69375 CDP45J 57390517 IC50 = 130 nM T69375 C28LIB 57390518 IC50 = 46 nM T69375 C8DZ1N 57390519 IC50 = 10 nM T69375 C7K4LJ 57390520 IC50 = 240 nM T69375 CG51FX 57392289 IC50 = 26 nM T69375 C2IZ3W 57392739 IC50 = 10 nM T69375 C9P1SC 57393560 IC50 = 11 nM T69375 CVH4X0 57394043 IC50 = 14 nM T69375 C1EYU6 57394468 IC50 = 38 nM T69375 CV9W8C 57395293 IC50 = 22 nM T69375 CQ2A1B 57395802 IC50 = 52 nM T69375 CW7XA9 57397040 IC50 = 9 nM T69375 C8FQH3 57402785 IC50 = 800 nM T69375 C6UAN1 57467725 IC50 = 1476 nM T69375 C7I4QD 57519510 IC50 = 283 nM T69375 CY8HG6 58017084 IC50 = 66 nM T69375 CO57NK 58155042 IC50 = 2070 nM T69375 CXJ63M 59603829 IC50 = 1700 nM T69375 CQEU96 59603842 IC50 = 640 nM T69375 C5IN0E 59718933 IC50 = 76 nM T69375 C5CO0X 59718937 IC50 = 390 nM T69375 C1XCV6 59718972 IC50 = 400 nM T69375 C20CME 59743327 IC50 = 24 nM T69375 C4IM1V 59743368 IC50 = 51 nM T69375 C6VYE9 59743400 IC50 = 151 nM T69375 CJE42G 59743404 IC50 = 1200 nM T69375 CUW7J8 59743407 IC50 = 21 nM T69375 C8L4KY 59743442 IC50 = 139 nM T69375 CSK8O7 59743445 IC50 = 57 nM T69375 C0MO4E 59743458 IC50 = 79 nM T69375 C5UYK1 59743461 IC50 = 64 nM T69375 CWB21E 59743477 IC50 = 246 nM T69375 C5RH4P 59743505 IC50 = 28 nM T69375 C3KY7N 59743507 IC50 = 47 nM T69375 CJ2NM1 59743549 IC50 = 194 nM T69375 CY89OP 59743571 IC50 = 27 nM T69375 C3J7CS 59846155 IC50 = 960 nM T69375 C2RCA7 59846164 IC50 = 900 nM T69375 CDA46Z 59846170 IC50 = 140 nM T69375 C86QAW 59846186 IC50 = 219 nM T69375 C20GMT 59846188 IC50 = 70 nM T69375 C5OL1V 59846192 IC50 = 1310 nM T69375 CTW8X2 59846211 IC50 = 507 nM T69375 C24GXO 59846214 IC50 = 220 nM T69375 CT0K1G 59846217 IC50 = 535 nM T69375 CFPS65 59846262 IC50 = 200 nM T69375 CMZU27 59846267 IC50 = 170 nM T69375 CG3WZ7 59846277 IC50 = 94 nM T69375 CO8R0G 59846284 IC50 = 32 nM T69375 C1MR8Q 60097495 IC50 > 10000 nM T69375 CVZ67M 66816803 IC50 = 64 nM T69375 CLG56W 66940332 IC50 = 86 nM T69375 C06UMH 66958119 IC50 = 806 nM T69375 C37NKO 67129970 IC50 > 10000 nM T69375 CK80LJ 67130050 IC50 > 10000 nM T69375 CV63UL 67240318 IC50 > 10000 nM T69375 CAWC35 68621678 IC50 > 1000 nM T69375 C7GRV2 68755406 IC50 > 10000 nM T69375 C5DGR9 69036886 IC50 = 10000 nM T69375 C51IQP 69309404 IC50 = 2900 nM T69375 CQ8HE2 70690944 IC50 > 30000 nM T69375 C13FWG 70695135 IC50 > 30000 nM T69375 C0VZB2 70697173 IC50 > 30000 nM T69375 CJ1SW3 71452229 IC50 = 3800 nM T69375 CF7N8W 71454040 IC50 = 87 nM T69375 CKT60L 71455860 Ki = 262 nM T69375 CU0EG4 71457558 IC50 = 190 nM T69375 CAK95D 71461189 IC50 = 290 nM T69375 C1DM6U 71461190 IC50 > 20000 nM T69375 CG0LC3 71654859 IC50 = 650 nM T69375 CHGS02 71654860 IC50 = 280 nM T69375 CTL1H9 71655707 IC50 = 35 nM T69375 C7OQC1 71720177 IC50 = 2180 nM T69375 CU9ZM5 72164196 IC50 = 100 nM T69375 CN8W3X 72164198 IC50 = 135 nM T69375 CQC51G 72164439 IC50 > 190 nM T69375 CI8CA4 72164562 IC50 > 190 nM T69375 CZ4BX1 72547959 IC50 = 514 nM T69375 CFSI04 72700746 IC50 = 120 nM T69375 CE2Y0X 73386882 IC50 = 220 nM T69375 C54KDR 86763302 IC50 = 311 nM T69375 C4HKT5 87057579 IC50 = 2836 nM T69375 C1HW4B 89735655 IC50 = 4400 nM T69375 CQ2OB9 90292687 IC50 > 10000 nM T69375 CHI39S 90292823 IC50 > 10000 nM T69375 C5C9PB 90667115 IC50 = 603 nM T69375 CI4RH8 90667116 IC50 = 1040 nM T69375 C4H0ZN 90667117 IC50 = 1440 nM T69375 CTB63D 90667118 IC50 = 3320 nM T69375 C5TPF3 90667119 IC50 = 860 nM T69375 C80FXC 90667121 IC50 = 329 nM T69375 C0HL7F 90667127 IC50 = 1410 nM T69375 C6FRO8 90667128 IC50 = 603 nM T69375 CE0ID8 90667129 IC50 = 1040 nM T69375 CZ45HF 90667130 IC50 = 2070 nM T69375 CSJ4C2 90667131 IC50 = 806 nM T69375 CJU4V7 90667132 IC50 = 1440 nM T69375 CBZ73T 90667133 IC50 = 3320 nM T69375 CW3UI2 90667134 IC50 = 860 nM T69375 C0M3VU 90667135 IC50 = 1 nM T69375 CH7G1F 90667136 IC50 = 1 nM T69375 C7P8TV 90667137 IC50 = 3 nM T69375 CE05TI 90667138 IC50 = 0.6 nM T69375 CH4DI3 90667139 IC50 = 0.68 nM T69375 C1U9DY 90667140 IC50 = 0.69 nM T69375 C9JQE0 90667141 IC50 = 0.51 nM T69375 CIV0J1 90667142 IC50 = 2.5 nM T69375 C1C7PW 90667143 IC50 = 0.71 nM T69375 CLF96U 90667144 IC50 = 34 nM T69375 C49JZU 90667145 IC50 = 0.24 nM T69375 C7V8BN 91754589 IC50 = 12 nM T69375 CQ2G3S 91754590 IC50 = 66 nM T69375 CJQ5N6 91936970 IC50 = 5000 nM T69375 C2GNI5 101891709 IC50 = 210 nM T69375 C61FOL 118144367 IC50 = 158 nM T69375 CY82JT 118146747 IC50 = 26 nM T69375 CIDU81 118146748 IC50 = 561 nM T69375 C8TLS2 118146764 IC50 = 463 nM T69375 CERD34 118146805 IC50 = 66 nM T69375 CJ4Z3K 118146817 IC50 = 3450 nM T69375 C7Q6RW 118146819 IC50 = 160 nM T69375 C4P9AK 118146855 IC50 = 148 nM T69375 CET9N4 118146870 IC50 = 29 nM T69375 C4PBE7 118146871 IC50 = 114 nM T69375 CNI34V 118146882 IC50 = 25 nM T69375 C8K0GC 118146884 IC50 = 428 nM T69375 C4O6MA 118146892 IC50 = 18 nM T69375 CR9ML7 118725554 IC50 = 336 nM T69375 CRUE70 122178088 IC50 = 241 nM T69375 CMG2E7 122178091 IC50 = 65 nM T69375 CQ0F5Z 122178092 IC50 = 434 nM T69375 C0FM1R 130196825 IC50 = 305 nM T69375 CA0ZK8 135499374 IC50 = 630 nM T69375 CTJ48K 135524085 IC50 = 240 nM T69375 CUT1W7 135524168 IC50 = 950 nM T69375 CM3UC9 135883136 IC50 > 100000 nM T69375 CP3LQ9 135890414 IC50 = 2 nM T69375 CZ5UN7 135890420 IC50 = 85 nM T69375 CV3E0X 135890430 IC50 = 22 nM T69375 C0OM5P 135890431 IC50 = 34 nM T69375 CP1Y5C 135890437 IC50 = 980 nM T69375 CH26QS 135890446 IC50 = 76 nM T69375 CM2UH4 135894362 IC50 > 1000 nM T69375 CY19DW 135894364 IC50 > 1000 nM T69375 C6T3QE 136025993 IC50 = 700 nM T69375 C6V5FC 136079665 IC50 = 198 nM T69375 CGX6C4 136173253 IC50 > 10000 nM T69375 C15HQK 136218656 IC50 > 1000 nM T69375 CZ06UK 136218660 IC50 > 1000 nM T69375 CML48X 136218661 IC50 > 1000 nM T69375 COB69I 136218662 IC50 > 1000 nM T69375 CSL6Q8 136218663 IC50 > 1000 nM T69375 CTFJ83 136226213 IC50 > 1000 nM T69375 C5EV8A 136240902 IC50 > 1000 nM T69375 CX9LB5 136240903 IC50 > 1000 nM T69375 CMC58H 136240944 IC50 > 1000 nM T69375 C60PRZ 136241012 IC50 > 1000 nM T69375 C1Q9YN 136252259 IC50 > 1000 nM T69375 CI1E8V 137634241 IC50 > 10000 nM T69375 CZ9BN4 138320062 IC50 = 0.059 nM T69375 C6VB3O 145925651 IC50 >= 5000 nM T69375 CFV10S 155529132 IC50 = 710 nM T69375 D00HVA 11624601 Ki = 4 nM T69375 D02PVB 8515 IC50 = 40 nM T69375 D07OXC 11650194 IC50 > 100000 nM T69375 D08LYB 5166 IC50 = 5 nM T69375 D0E8KF 824661 IC50 > 10000 nM T69375 D0EW9J 10389239 IC50 > 200000 nM T69375 D0F5BY 11507052 IC50 = 4663 nM T69375 D0L0HG 766949 IC50 = 316.23 nM T69375 D0OZ2S 11785878 IC50 > 40000 nM T69375 D0Q3NG 11715520 IC50 = 1100 nM T69375 D0QN6U 9806182 IC50 = 2200 nM T69375 D0S7IE 11658882 IC50 = 7700 nM T69375 D0VJ2S 57340686 IC50 = 1 nM T75243 D06OMK 445643 IC50 = 3.162 nM T75243 D09XZB 123631 IC50 > 50000 nM T75243 D0B3HD 2519 IC50 = 400000 nM T75243 D0E6XR 3062316 IC50 = 35000 nM T75243 D0ES1Q 6918289 IC50 = 1760 nM T75243 D0J5VR 11625818 IC50 > 1000 nM T75243 D0R0MW 5329102 IC50 > 50000 nM T75243 D0S5LD 135565596 IC50 = 45 nM T75243 D0V7WS 9876378 IC50 = 3.3 nM T75243 D0W5HK 216239 IC50 > 50000 nM T75243 D01PGR 16123056 IC50 = 157 nM T75243 D01QSO 16654980 IC50 = 94 nM T75243 D03DPZ 45375953 Ki = 1 nM T75243 D03EZE 25167777 IC50 = 0.31 nM T75243 D03LWG 53235510 IC50 > 10000 nM T75243 D03XAQ 49784945 IC50 = 1600 nM T75243 D05EXN 58298316 IC50 = 10 nM T75243 D07BGC 57384863 Ki = 70 nM T75243 D07EHV 44814409 IC50 > 9100 nM T75243 D08QGT 17755052 IC50 = 3 nM T75243 D0AW5T 9849735 IC50 = 3100 nM T75243 D0D8JB 44516953 IC50 = 0.4 nM T75243 D0E6UZ 54575456 IC50 = 431 nM T75243 D0H9DA 54761306 IC50 = 370 nM T75243 D0N5JZ 25033539 IC50 = 7.9 nM T75243 D0O1IM 58298318 IC50 = 21 nM T75243 D0O1LD 11647372 IC50 = 350 nM T75243 D0O6VZ 25254071 Ki = 17 nM T75243 D0TU7B 58507717 Ki = 62 nM T75243 D0U8QH 59239165 Ki = 3.8 nM T75243 D0UP1Z 51001932 Ki = 1200 nM T75243 D0VG0D 11977753 IC50 = 5 nM T75243 D0W7HE 56649450 IC50 > 9100 nM T75243 D0XD4I 118502708 IC50 = 200 nM T75243 D0Z2UQ 25262792 IC50 = 2.8 nM T75243 D04PGB 445501 IC50 = 20892.96 nM T75243 D05HIJ 135565159 IC50 > 10000 nM T75243 D09SFV 3973 IC50 = 2500 nM T75243 D0K1VK 25262965 IC50 = 4 nM T75243 D0P1JI 312145 IC50 = 40 nM T75243 D0U2TQ 644215 IC50 = 800 nM T75243 CB1VW3 1400 IC50 = 9318 nM T75243 CH5QF8 1018277 IC50 = 570 nM T75243 CRGP15 1420707 IC50 = 52200 nM T75243 CT2VP9 1471775 IC50 = 1410 nM T75243 C9LG0N 1476679 IC50 = 5000 nM T75243 C49EKU 1862374 IC50 = 8300 nM T75243 C0NMD8 1882360 IC50 = 57600 nM T75243 C7CSH6 2024268 IC50 = 32200 nM T75243 CQ02GR 2930286 IC50 = 54100 nM T75243 C6T0BZ 4899677 IC50 = 20400 nM T75243 C4G6WY 5253082 IC50 > 2000 nM T75243 CZ7GL8 9809998 IC50 = 9.6 nM T75243 CNQJ46 9867340 IC50 = 193 nM T75243 CJ79RC 9879653 IC50 = 37 nM T75243 C7HMO6 11526786 IC50 = 2920 nM T75243 CFZO21 11979157 IC50 = 2 nM T75243 CBZU35 11997784 IC50 = 460 nM T75243 CEBI25 12050235 IC50 < 10000 nM T75243 CJCG06 12050236 IC50 < 10000 nM T75243 C0KX2Q 12050237 IC50 < 10000 nM T75243 C2DS5Z 12050238 IC50 < 10000 nM T75243 C63PLZ 12050239 IC50 < 10000 nM T75243 CZ7UR5 12050240 IC50 < 10000 nM T75243 CV9US5 16736978 IC50 = 3 nM T75243 C59CVU 19689599 IC50 > 20000 nM T75243 CTF23G 20644743 IC50 > 50000 nM T75243 CZ7V8L 21048651 IC50 > 50000 nM T75243 C0EJK3 23585071 IC50 = 288.4 nM T75243 CEYL29 23585510 IC50 > 9100 nM T75243 CBL37C 23642173 IC50 > 9100 nM T75243 C0EKO5 24772654 IC50 > 10000 nM T75243 CBS5J4 24804985 IC50 = 28 nM T75243 C9PA0M 24807809 IC50 = 28600 nM T75243 C5E4QN 24807810 IC50 > 20000 nM T75243 C3QKS1 24807976 IC50 = 5600 nM T75243 CGJ60P 24807978 IC50 = 14000 nM T75243 CIPF03 24808145 IC50 > 20000 nM T75243 C2XLC5 24808146 IC50 > 20000 nM T75243 C7DX6N 24808147 IC50 = 6500 nM T75243 CY61FQ 24808148 IC50 = 8700 nM T75243 C72QHP 24808149 IC50 > 20000 nM T75243 CBMA95 24808336 IC50 > 20000 nM T75243 C7FD1B 24808337 IC50 > 20000 nM T75243 CCP2M3 24822704 IC50 > 50000 nM T75243 CB79YC 24905143 IC50 = 2100 nM T75243 C2DC9J 24905144 IC50 = 100000 nM T75243 CN6V8Z 24905145 IC50 = 72 nM T75243 CSB7P5 24905148 IC50 = 4800 nM T75243 CGSF21 24905149 IC50 = 50000 nM T75243 CVDG02 24905150 IC50 > 50000 nM T75243 CWH6C5 24905152 IC50 = 140 nM T75243 C0HE2Q 24905153 IC50 = 1700 nM T75243 C7QSC9 24905154 IC50 = 80 nM T75243 CO9D0K 24905155 IC50 = 100000 nM T75243 C5W9UR 24905157 IC50 = 934 nM T75243 CC1DA3 24905158 IC50 = 766 nM T75243 COW79F 24905159 IC50 = 5000 nM T75243 CFPA53 24905160 IC50 = 40000 nM T75243 C2O0JX 24905161 IC50 = 3800 nM T75243 CA72BE 24905162 IC50 = 4300 nM T75243 CQN6X9 24905163 IC50 = 4500 nM T75243 CD4O1F 24905165 IC50 = 100000 nM T75243 CKL48T 24905166 IC50 = 3500 nM T75243 C76VYL 24905167 IC50 = 12000 nM T75243 C7K5PU 24905168 IC50 = 4300 nM T75243 CZ57ID 24905169 IC50 = 8000 nM T75243 C2DHX9 24905170 IC50 = 5500 nM T75243 CSB96E 24905171 IC50 = 50000 nM T75243 CWZ0R2 24905172 IC50 = 1900 nM T75243 CY3B6M 24905175 IC50 = 8200 nM T75243 CW7UA3 24905176 IC50 = 404 nM T75243 CW1V0H 24905177 IC50 = 100000 nM T75243 CO6Y0L 24905178 IC50 = 5500 nM T75243 C60NQW 24905179 IC50 = 635 nM T75243 C4MO8B 24905180 IC50 = 192 nM T75243 COJI47 24905181 IC50 = 692 nM T75243 CS0B2C 24905182 IC50 = 10000 nM T75243 C1H4BT 24905183 IC50 = 1900 nM T75243 C4WHK9 24905184 IC50 = 10000 nM T75243 C7Q4MZ 24905185 IC50 = 300 nM T75243 CS4IP1 24905186 IC50 = 30000 nM T75243 C69QWO 24905187 IC50 = 576 nM T75243 C85ANB 24905188 IC50 = 364 nM T75243 CNHD75 24905189 IC50 = 2500 nM T75243 C9JUO2 24905190 IC50 = 8000 nM T75243 CPR03K 24905191 IC50 = 5400 nM T75243 CTAG19 24905193 IC50 = 407 nM T75243 C7VJM5 24905194 IC50 = 4500 nM T75243 CEP1L3 24905195 IC50 = 3400 nM T75243 CP68ZD 24905196 IC50 = 1600 nM T75243 C8Z0RJ 24905197 IC50 = 110 nM T75243 CN9RT0 24905198 IC50 = 18000 nM T75243 CHI78P 24905200 IC50 = 1900 nM T75243 CO6PE8 24905201 IC50 = 467 nM T75243 CZ63HS 24905202 IC50 = 60 nM T75243 C2X0FC 24905203 IC50 = 1200 nM T75243 C0WCE3 24905204 IC50 = 3000 nM T75243 CNK50B 24905205 IC50 = 550 nM T75243 C12DPB 24905206 IC50 = 596 nM T75243 C8N0RH 24905207 IC50 = 100000 nM T75243 CYA5G2 24905208 IC50 = 565 nM T75243 CDV2B4 24905209 IC50 = 8300 nM T75243 CEFK68 24905210 IC50 = 412 nM T75243 CUFP12 24905211 IC50 = 243 nM T75243 C0JG8L 24905212 IC50 = 493 nM T75243 CQ13ZI 24905215 IC50 = 2200 nM T75243 C6VI8F 24905216 IC50 = 113 nM T75243 CXNH25 24905217 IC50 = 1500 nM T75243 C2PN9S 24905218 IC50 = 632 nM T75243 C9O2AL 24905219 IC50 = 1100 nM T75243 CIT7U8 24905220 IC50 = 2200 nM T75243 CMD26S 24905221 IC50 = 457 nM T75243 C4R8WC 24905222 IC50 = 205 nM T75243 C47SHA 24905223 IC50 = 657 nM T75243 C1DY2R 24905224 IC50 = 1100 nM T75243 CS0XF9 24905225 IC50 = 6800 nM T75243 CG5VX2 24905226 IC50 = 8700 nM T75243 C57QEO 24905227 IC50 = 100000 nM T75243 C7CG5E 24905228 IC50 = 783 nM T75243 CHP5D1 24905229 IC50 = 1300 nM T75243 CXP09S 24905230 IC50 = 426 nM T75243 CY7XG1 24905231 IC50 = 3200 nM T75243 C7JFQ2 24905232 IC50 = 33 nM T75243 C2JM1P 24905233 IC50 = 10000 nM T75243 CC3BF0 24905234 IC50 = 100000 nM T75243 CE57FI 24905235 IC50 = 30000 nM T75243 CUP20O 24905236 IC50 = 100000 nM T75243 CLC6Q2 24905237 IC50 = 100000 nM T75243 C9M1GI 24905238 IC50 = 2400 nM T75243 CVD72F 24905239 IC50 = 1640 nM T75243 CK38IZ 24905240 IC50 = 596 nM T75243 CO2V5E 24905241 IC50 = 3600 nM T75243 CZBA19 24905244 IC50 = 7000 nM T75243 CQ8OI1 24905246 IC50 = 7600 nM T75243 CIF2J5 24905251 IC50 = 100000 nM T75243 CPTE58 24905252 IC50 = 3600 nM T75243 CP50RD 24905280 IC50 = 37 nM T75243 CG13ZM 24905281 IC50 = 911 nM T75243 CF0S6X 24905282 IC50 = 3300 nM T75243 C5HBL0 24905284 IC50 = 1200 nM T75243 C2Z5DN 24905285 IC50 = 4000 nM T75243 CL6GH8 24905286 IC50 = 710 nM T75243 CKYO98 24905287 IC50 = 33 nM T75243 CRNQ65 24905288 IC50 = 3 nM T75243 COD7I5 24905289 IC50 = 16 nM T75243 C4LP7E 24905290 IC50 = 861 nM T75243 CE9JC2 24905291 IC50 = 98 nM T75243 C2GI1R 24905292 IC50 = 100000 nM T75243 CHW8C4 24905293 IC50 = 20 nM T75243 CQF0H1 24905294 IC50 = 40 nM T75243 CNO7X0 24905295 IC50 = 130 nM T75243 C5WRG7 24905296 IC50 = 6500 nM T75243 CQ1S0U 24905297 IC50 = 4800 nM T75243 C4UES7 24905298 IC50 = 616 nM T75243 CMS69P 24905299 IC50 = 3200 nM T75243 CC0U5M 24905300 IC50 = 439 nM T75243 CW7X6S 24905301 IC50 = 100000 nM T75243 C97IQV 24905302 IC50 = 1800 nM T75243 CSJ47V 24905303 IC50 = 3000 nM T75243 CPN74C 24905304 IC50 = 15000 nM T75243 C5CS3N 24905305 IC50 = 4800 nM T75243 CK4XE9 24905307 IC50 = 50000 nM T75243 CTU6Z3 24905308 IC50 = 100000 nM T75243 C9SQX1 24905309 IC50 = 6500 nM T75243 CM75JP 24905310 IC50 = 5000 nM T75243 C9Q2BJ 24905311 IC50 = 3900 nM T75243 C9VUA1 24905312 IC50 = 2400 nM T75243 CU3RS1 24905313 IC50 = 5100 nM T75243 CYG3H2 24905314 IC50 = 30000 nM T75243 CV5Q7O 24905315 IC50 = 815 nM T75243 C8SA3O 24905316 IC50 = 170 nM T75243 CI5MN3 24905317 IC50 = 377 nM T75243 CJ1P7K 24905318 IC50 = 450 nM T75243 C1T6YQ 24905319 IC50 = 9200 nM T75243 CAU86X 24905320 IC50 = 1000 nM T75243 C54ISY 24905321 IC50 = 11000 nM T75243 C2GE5I 24905322 IC50 = 2000 nM T75243 C8D6YK 24905323 IC50 = 2900 nM T75243 C5NZH9 24905324 IC50 = 880 nM T75243 C9D6JR 24905325 IC50 = 1500 nM T75243 CLZT41 24905326 IC50 = 230 nM T75243 CW8FD3 24905327 IC50 = 1100 nM T75243 CHB7A2 24905328 IC50 = 2200 nM T75243 CA8EI3 24905329 IC50 = 833 nM T75243 CCQ0O7 24905330 IC50 = 100000 nM T75243 CJ81AS 24905331 IC50 = 548 nM T75243 C8PW4H 24905332 IC50 = 127 nM T75243 C2Y5TF 24905333 IC50 = 156 nM T75243 CH9FL5 24905334 IC50 = 1200 nM T75243 C1S0PC 24905335 IC50 = 1700 nM T75243 C8N9MV 24905336 IC50 = 1100 nM T75243 C9E8BJ 24905338 IC50 = 5000 nM T75243 CX85AC 24905341 IC50 = 5800 nM T75243 CKZ80E 24905342 IC50 = 14000 nM T75243 CO8SH1 24905343 IC50 = 3100 nM T75243 C7IZL6 24905344 IC50 = 5400 nM T75243 C3IYB2 24936050 IC50 = 0.08 nM T75243 CLD3X6 24936051 IC50 = 620 nM T75243 C98MEW 24946175 IC50 = 17 nM T75243 CC7H3U 24946706 IC50 = 880 nM T75243 CD5HQ0 24969301 IC50 > 10000 nM T75243 CCZO17 24970164 IC50 = 130 nM T75243 CXI65T 24983588 IC50 = 64 nM T75243 CH6Q7Y 24983749 IC50 = 176 nM T75243 C6Q8HD 24983903 IC50 = 273 nM T75243 C7NYZ4 24984057 IC50 = 231 nM T75243 CV79PK 24984058 IC50 = 21 nM T75243 CX24TD 24985362 IC50 = 60 nM T75243 CV5OB6 24985365 IC50 = 190 nM T75243 CBGM96 24985541 IC50 = 580 nM T75243 C2DLE6 24985542 IC50 > 10000 nM T75243 CORB97 24985709 IC50 = 1690 nM T75243 CQ39PB 24985717 IC50 = 5 nM T75243 C0G9DN 24985874 IC50 = 1360 nM T75243 CGSE92 25009673 Ki = 911 nM T75243 CB7VT5 25032306 Ki = 11.1 nM T75243 C2H3WJ 25032388 Ki = 2.54 nM T75243 C17PCM 25032389 Ki = 4.52 nM T75243 CM1GB6 25032390 Ki = 92.6 nM T75243 C0W2TF 25032391 Ki = 8.8 nM T75243 CCR6S7 25032392 Ki = 9.1 nM T75243 CBU2H9 25032644 Ki = 17 nM T75243 CHR51O 25057242 IC50 = 1800 nM T75243 C0T4NK 25070551 IC50 = 7200 nM T75243 C1UKQ4 25070552 IC50 = 2100 nM T75243 CZRA03 25070553 IC50 = 600 nM T75243 CO20FT 25070554 IC50 = 140 nM T75243 CL4B5Z 25070555 IC50 = 10500 nM T75243 C7U0SC 25070882 IC50 = 634 nM T75243 CCN36H 25071204 IC50 = 970 nM T75243 CQ7P4X 25071206 IC50 = 160 nM T75243 C14SFA 25071208 IC50 = 590 nM T75243 CNCJ40 25071516 IC50 = 570 nM T75243 CXWO13 25071518 IC50 = 310 nM T75243 CBH13R 25071519 IC50 = 160 nM T75243 CJM7O0 25071520 IC50 = 1700 nM T75243 C68PFD 25073081 IC50 = 170 nM T75243 CBJ20X 25073385 IC50 = 51 nM T75243 CZN7W0 25073388 IC50 = 152 nM T75243 C8DG4R 25109014 Ki = 59 nM T75243 CB3W1F 25109202 Ki = 42 nM T75243 CTO19H 25109378 Ki = 10 nM T75243 C83WVR 25109494 Ki = 30 nM T75243 CK2YI4 25168990 IC50 = 1.514 nM T75243 CC1D8V 25172062 IC50 = 300 nM T75243 CPW2D9 25172477 IC50 = 234 nM T75243 CXG59Q 25175568 IC50 = 303 nM T75243 C1C9ZF 25182020 IC50 = 913 nM T75243 CUA41N 25182022 IC50 > 6000 nM T75243 CX2N5M 25182023 IC50 > 6000 nM T75243 C46ZAW 25182142 IC50 > 6000 nM T75243 CP17FV 25182145 IC50 > 6000 nM T75243 CGQ56K 25182146 IC50 > 6000 nM T75243 C9G6DH 25182281 IC50 = 3010 nM T75243 CS07FL 25182282 IC50 > 6000 nM T75243 C2LYI1 25182285 IC50 > 6000 nM T75243 C7GAR5 25182286 IC50 > 6000 nM T75243 C9X3OT 25182424 IC50 > 6000 nM T75243 C0JBX1 25182427 IC50 > 6000 nM T75243 CAG4R1 25182562 IC50 > 6000 nM T75243 C5JD1M 25182565 IC50 > 6000 nM T75243 CWIH67 25182709 IC50 > 6000 nM T75243 C6O1VG 25182710 IC50 > 6000 nM T75243 C80UYN 25182711 IC50 > 6000 nM T75243 C8H9ET 25182714 IC50 > 6000 nM T75243 CD8M0G 25182867 IC50 > 6000 nM T75243 C9T6AZ 25182868 IC50 > 6000 nM T75243 C0S4YF 25182871 IC50 > 6000 nM T75243 CS4N6U 25183031 IC50 > 6000 nM T75243 CX8F3W 25183032 IC50 > 6000 nM T75243 C38MPQ 25195571 IC50 = 4.8 nM T75243 C1CL7V 25195572 IC50 = 2.4 nM T75243 CD4L2F 25195682 IC50 = 0.8 nM T75243 C4QTX9 25195788 IC50 = 0.3 nM T75243 CIRE40 25195789 IC50 = 23 nM T75243 CHJM38 25195893 IC50 = 65 nM T75243 C64SIJ 25195997 IC50 = 125 nM T75243 CB6CP3 25196219 IC50 = 16 nM T75243 CWN52I 25196221 IC50 = 1.4 nM T75243 C8RWY2 25196900 IC50 = 120 nM T75243 CNU28R 25197239 IC50 = 2.7 nM T75243 CMST49 25197240 IC50 = 0.8 nM T75243 CLW96O 25207689 Ki = 21 nM T75243 CRO09K 25211064 IC50 > 30000 nM T75243 C6MR3O 25229450 IC50 = 4.6 nM T75243 CQL23A 25229526 IC50 = 9 nM T75243 CWP29U 25242324 Ki = 30 nM T75243 C58WEU 25260757 IC50 = 0.21 nM T75243 C9V5KO 25260758 IC50 = 0.22 nM T75243 C8RYX7 25260759 IC50 = 0.24 nM T75243 C47RYE 25260913 IC50 = 0.19 nM T75243 C96OGS 25260915 IC50 = 0.38 nM T75243 CBCF51 25261227 IC50 = 0.5 nM T75243 C5DQF0 25261230 IC50 = 0.19 nM T75243 C4V2EJ 25261231 IC50 = 0.46 nM T75243 C3I9SN 25261388 IC50 = 0.23 nM T75243 C7SNP6 25261389 IC50 = 0.22 nM T75243 C4R3ZS 25261390 IC50 = 0.26 nM T75243 CUR93V 25261554 IC50 = 0.62 nM T75243 CCR83Z 25261555 IC50 = 0.11 nM T75243 C38UOX 25262174 IC50 = 0.48 nM T75243 CD27XK 25262616 IC50 = 0.74 nM T75243 CPLM23 25262617 IC50 = 0.6 nM T75243 CU6C8J 25262782 IC50 = 0.3 nM T75243 CT97DF 25262783 IC50 = 0.1 nM T75243 CFL6G2 25262946 IC50 = 1.34 nM T75243 CO4PL8 42606076 IC50 = 5100 nM T75243 C20VGT 42606077 IC50 = 10700 nM T75243 C7N5EC 42606078 IC50 = 10800 nM T75243 CI69YO 42606079 IC50 > 100000 nM T75243 C5L7IT 42606080 IC50 > 50000 nM T75243 CG04LZ 42606083 IC50 > 100000 nM T75243 C0WEU1 42606190 IC50 > 100000 nM T75243 CD6LN3 42606191 IC50 > 50000 nM T75243 CWR7P5 42606194 IC50 > 50000 nM T75243 CJ2GM1 42606195 IC50 > 50000 nM T75243 C61JUL 42606196 IC50 > 50000 nM T75243 C9GS8P 42606431 IC50 = 19100 nM T75243 CW63VM 42609338 Ki = 30 nM T75243 CYJK74 42632991 IC50 = 5900 nM T75243 CQW60S 42632992 IC50 = 3650 nM T75243 C2FIY7 42633175 IC50 = 2000 nM T75243 CL2XD7 42633904 IC50 > 4000 nM T75243 C9B0DZ 42633906 IC50 > 4000 nM T75243 CHP49D 42635321 IC50 = 355 nM T75243 C96ETP 42635322 IC50 = 1625 nM T75243 CZN3G1 42635323 IC50 = 5000 nM T75243 CCV0R1 42635502 IC50 = 430 nM T75243 CR8C3W 42635504 IC50 = 3600 nM T75243 C10RBA 42636535 IC50 > 5000 nM T75243 C3ROX1 44124863 IC50 = 0.4 nM T75243 C2YQX8 44125256 IC50 = 35 nM T75243 CV5O8L 44125375 IC50 = 20 nM T75243 C5JN4O 44125376 IC50 = 20 nM T75243 C0U2OY 44125377 IC50 = 6.6 nM T75243 C5CQK3 44138092 IC50 = 1 nM T75243 CP61GU 44156032 IC50 = 18 nM T75243 C3CBU7 44156033 IC50 = 500 nM T75243 C7XI2W 44156156 IC50 = 2 nM T75243 C63BLR 44156157 IC50 = 1 nM T75243 C19LGE 44158465 IC50 = 420 nM T75243 CG4DY5 44158569 IC50 = 95 nM T75243 CB46RQ 44159380 IC50 = 96 nM T75243 CIKM57 44180156 IC50 = 289 nM T75243 CXL61J 44181600 IC50 = 610 nM T75243 CO0YZ7 44182308 IC50 = 0.83 nM T75243 CS0M9A 44187604 IC50 = 0.63 nM T75243 C0BRI9 44187779 IC50 = 21 nM T75243 CDA81B 44187783 IC50 = 0.89 nM T75243 C0LB8S 44187784 IC50 = 3 nM T75243 CCTO21 44187951 IC50 = 2.55 nM T75243 CVYS60 44187952 IC50 = 0.5 nM T75243 C8X3UZ 44187955 IC50 = 2.2 nM T75243 CJU85Z 44188321 IC50 = 2.7 nM T75243 CHU02A 44188322 IC50 = 0.56 nM T75243 C69HQS 44188840 IC50 = 0.84 nM T75243 CD78AG 44188841 IC50 = 3.05 nM T75243 CY7EL1 44188842 IC50 = 0.51 nM T75243 C0SE1X 44188843 IC50 = 0.57 nM T75243 CG13ZF 44188844 IC50 = 0.32 nM T75243 CR0BF9 44189010 IC50 = 0.35 nM T75243 C71NFL 44189011 IC50 = 1.6 nM T75243 C39ABJ 44189192 IC50 = 0.31 nM T75243 CK73NR 44219749 IC50 = 4.3 nM T75243 C2V6WY 44232672 IC50 = 9.6 nM T75243 CA91IW 44232914 IC50 = 7 nM T75243 CN10TK 44232915 IC50 = 2450 nM T75243 CNY95J 44232916 IC50 = 46 nM T75243 COXT27 44232917 IC50 = 1.5 nM T75243 CFC2A1 44232918 IC50 = 1.4 nM T75243 CVN7P2 44233160 IC50 = 0.52 nM T75243 CQXD21 44233161 IC50 = 22 nM T75243 CI7N6F 44233162 IC50 = 2.1 nM T75243 CC6H5K 44233163 IC50 = 2 nM T75243 CSGQ48 44233164 IC50 = 1.1 nM T75243 CI65AN 44233388 IC50 = 1 nM T75243 CS9UA8 44233389 IC50 = 0.32 nM T75243 CZ3L7W 44233390 IC50 = 0.6 nM T75243 CA7R1U 44233391 IC50 = 0.5 nM T75243 CN4A7W 44233639 IC50 = 0.2 nM T75243 CWLA98 44233640 IC50 = 0.3 nM T75243 CXO1L7 44233641 IC50 = 0.34 nM T75243 CX7B1Y 44264159 IC50 < 10000 nM T75243 CVM4J9 44264177 IC50 < 10000 nM T75243 C8RNS0 44264540 IC50 < 10000 nM T75243 CA45LZ 44396556 IC50 = 1.45 nM T75243 C5EYH7 44396557 IC50 = 1.88 nM T75243 C52ZQN 44405685 IC50 = 5.8 nM T75243 C4QG5B 44405767 IC50 = 4.8 nM T75243 C2QF1N 44457157 IC50 = 829 nM T75243 C34HLQ 44457158 IC50 = 692 nM T75243 CSW53V 44457165 IC50 = 961 nM T75243 CZ4O2K 44457166 IC50 = 820 nM T75243 C6JS1G 44457167 IC50 = 890 nM T75243 CW5KH3 44457168 IC50 = 1870 nM T75243 CCBP46 44457169 IC50 > 1690 nM T75243 CWTU20 44457172 IC50 > 18700 nM T75243 C2QR9D 44457173 IC50 = 12600 nM T75243 C9H2FA 44457174 IC50 = 13900 nM T75243 C9X8CD 44457178 IC50 = 1210 nM T75243 CD4RP9 44457179 IC50 = 1350 nM T75243 C16ASL 44457183 IC50 = 3560 nM T75243 CA04RG 44457184 IC50 = 2330 nM T75243 C8INQ7 44457185 IC50 = 2290 nM T75243 C0UBI8 44457188 IC50 = 767 nM T75243 CGCS67 44457189 IC50 = 1480 nM T75243 C9WG2B 44457191 IC50 = 3570 nM T75243 C4OK8P 44457192 IC50 = 878 nM T75243 CHSE37 44457195 IC50 = 1470 nM T75243 CN9H7F 44457201 IC50 = 1800 nM T75243 CI6G5C 44457211 IC50 = 960 nM T75243 C9N4PA 44457212 IC50 = 831 nM T75243 CB70NU 44457213 IC50 = 816 nM T75243 CY4H8C 44457218 IC50 = 568 nM T75243 C0RN9S 44457220 IC50 = 822 nM T75243 C2JV8Y 44457231 IC50 = 2450 nM T75243 CQD4T3 44457232 IC50 = 1690 nM T75243 CT02VO 44457235 IC50 = 249 nM T75243 CB2J6E 44457236 IC50 = 619 nM T75243 CG7YT9 44457237 IC50 = 1200 nM T75243 CVG75D 44473371 IC50 = 0.5 nM T75243 CX3FK1 44513884 IC50 = 1.2 nM T75243 CL4RO5 44513885 IC50 = 1.2 nM T75243 C6RC9J 44513886 IC50 = 3.9 nM T75243 CGS7Q4 44513887 IC50 = 1.7 nM T75243 CSVD32 44513888 IC50 = 6.3 nM T75243 CLN2M5 44514201 IC50 = 3.9 nM T75243 C2Y8ML 44514203 IC50 = 6.7 nM T75243 CA9H8D 44514205 IC50 = 9.3 nM T75243 C01ZJI 44514208 IC50 = 0.3 nM T75243 CZ8WK6 44514210 IC50 = 0.4 nM T75243 CI8H3K 44514481 IC50 = 10 nM T75243 C51SEJ 44515083 IC50 = 1.8 nM T75243 CXBV98 44515084 IC50 = 1.9 nM T75243 C73HNB 44515696 IC50 = 2.5 nM T75243 CB7XW5 44516307 IC50 = 1.5 nM T75243 C4W5EM 44516309 IC50 = 1.4 nM T75243 C8VAU1 44516310 IC50 = 0.7 nM T75243 C8I1ZB 44516311 IC50 = 0.6 nM T75243 CSJ95V 44516635 IC50 = 0.8 nM T75243 CV6Z0N 44516636 IC50 = 0.7 nM T75243 CB3MV8 44517288 IC50 = 1.3 nM T75243 CDEQ97 44520808 IC50 = 215 nM T75243 CT7DW6 44520809 IC50 = 49 nM T75243 C3T2YD 44520810 IC50 = 4 nM T75243 CJP71L 44520811 IC50 = 6 nM T75243 CB4RN0 44520812 IC50 = 83 nM T75243 CGQ1F8 44520814 IC50 = 695 nM T75243 C2W5QS 44520815 IC50 = 7300 nM T75243 CN78XU 44520816 IC50 = 5950 nM T75243 C1TI9F 44520817 IC50 = 190 nM T75243 CHS6C1 44520818 IC50 = 130 nM T75243 CKP60Q 44520819 IC50 = 145 nM T75243 C0XEA9 44520820 IC50 = 88 nM T75243 CFE63J 44520821 IC50 = 230 nM T75243 CV43BN 44520822 IC50 = 380 nM T75243 CYU2B5 44520824 IC50 = 170 nM T75243 C73ZYA 44520825 IC50 = 4 nM T75243 CB25DI 44539683 IC50 = 1.4 nM T75243 CNWO35 44539684 IC50 = 0.67 nM T75243 C8MTO3 44539685 IC50 = 7.5 nM T75243 CTQ06N 44539783 IC50 = 42 nM T75243 C3D8CF 44540543 IC50 = 0.46 nM T75243 C0Z3QI 44540642 IC50 = 37 nM T75243 C3Z7GL 44540644 IC50 = 0.94 nM T75243 CGB2A8 44540925 IC50 = 9.5 nM T75243 CFI4O2 44541101 IC50 = 11 nM T75243 CW19QS 44544943 Ki = 950 nM T75243 C6L4SV 44545041 Ki = 72 nM T75243 C0IX1C 44545849 IC50 = 3 nM T75243 C6HC3L 44548482 IC50 = 5.3 nM T75243 CH3L9P 44551660 IC50 = 4590 nM T75243 CYMD49 44552663 IC50 = 1650 nM T75243 C6B7LH 44552664 IC50 = 11 nM T75243 C3QZX0 44552666 IC50 = 18 nM T75243 C64OQC 44552667 IC50 = 9 nM T75243 C7LG6Q 44552844 IC50 = 118 nM T75243 C9T2CZ 44552845 IC50 = 18 nM T75243 CXLD75 44552846 IC50 = 108 nM T75243 CALT95 44554240 IC50 = 130 nM T75243 CVDA08 44554755 IC50 = 190 nM T75243 C25EGX 44554909 IC50 = 280 nM T75243 C6VR1P 44554910 IC50 = 123 nM T75243 CR4J0X 44554913 IC50 = 3700 nM T75243 CWV2T9 44554915 IC50 = 153 nM T75243 CCW12H 44555222 IC50 = 265 nM T75243 CTM8S9 44555225 IC50 = 2125 nM T75243 C7PSO6 44555226 IC50 = 430 nM T75243 C3VRO9 44557921 IC50 > 10000 nM T75243 C8A5RT 44577639 IC50 > 15000 nM T75243 C5VNA7 44599029 IC50 = 2 nM T75243 CCFX21 44599203 IC50 = 1 nM T75243 CU5YK1 44599206 IC50 = 1.7 nM T75243 C4OP3Y 44599690 IC50 = 0.6 nM T75243 C7H0XM 44599855 IC50 = 1.7 nM T75243 CL73YV 44600010 IC50 = 0.5 nM T75243 C54ZQB 44600166 IC50 = 0.9 nM T75243 C2ZYD0 44600649 IC50 = 0.4 nM T75243 C3R2PX 44600650 IC50 = 205 nM T75243 C8AT9I 44600651 IC50 = 64 nM T75243 C5JL6C 44600806 IC50 = 1 nM T75243 CJUQ51 44600808 IC50 > 800 nM T75243 C0BXS4 44600809 IC50 > 800 nM T75243 CA9LP4 44600952 IC50 = 3 nM T75243 CFK83C 44600954 IC50 = 7 nM T75243 CX30VY 44600955 IC50 = 2 nM T75243 C9N1SY 44600956 IC50 = 8 nM T75243 CUI9Y8 44601112 IC50 = 30 nM T75243 CBV38N 44601113 IC50 = 33 nM T75243 CA3K8E 44601278 IC50 = 7 nM T75243 CZX94G 44601279 IC50 = 52 nM T75243 CD1A2Z 44601448 IC50 = 11 nM T75243 CB12CS 44601449 IC50 = 24 nM T75243 CIDT64 44601450 IC50 = 14 nM T75243 CWY15L 44604823 IC50 = 2.6 nM T75243 CN9ZD0 44604824 IC50 = 0.7 nM T75243 CL3S1F 44604825 IC50 = 23 nM T75243 C28QLM 44605035 IC50 = 4.6 nM T75243 C75XHS 44605037 IC50 = 0.4 nM T75243 CFN95D 44605038 IC50 = 0.3 nM T75243 CD8Q9Z 44605039 IC50 = 0.1 nM T75243 CI70YP 44605246 IC50 = 0.7 nM T75243 C36ZFK 44605247 IC50 = 0.8 nM T75243 CEK25C 44605248 IC50 = 0.6 nM T75243 C3F4UX 44605249 IC50 = 0.2 nM T75243 CQ0FZ7 44605426 IC50 = 0.3 nM T75243 CC7G2L 44605427 IC50 = 0.5 nM T75243 CDLP04 44605428 IC50 = 0.7 nM T75243 CSKN09 44605429 IC50 = 0.5 nM T75243 CA79QG 44605430 IC50 = 0.6 nM T75243 CM49FO 44605789 IC50 = 2.3 nM T75243 C3DK5F 44605790 IC50 = 1.9 nM T75243 C9Z4TY 44605791 IC50 = 0.62 nM T75243 C9F8JY 44605792 IC50 = 0.87 nM T75243 CGT58A 44606131 IC50 = 0.6 nM T75243 CTO96K 44606133 IC50 = 0.23 nM T75243 CH7O9Y 44606302 IC50 = 1.2 nM T75243 C8Y4FE 44606303 IC50 = 0.58 nM T75243 C4PEO6 44606304 IC50 = 1 nM T75243 CG04KF 44606474 IC50 = 5.5 nM T75243 C86RYX 44606475 IC50 = 91 nM T75243 CNI9G3 44606476 IC50 = 1.9 nM T75243 CE90UX 44606477 IC50 = 53 nM T75243 CQIY50 44606640 IC50 = 17 nM T75243 C1ML5R 44606641 IC50 = 1.8 nM T75243 C35QOE 44606642 IC50 = 1.8 nM T75243 CWQ67K 44606643 IC50 = 1.2 nM T75243 CY0QH9 44606644 IC50 = 0.28 nM T75243 CFQT17 44606818 IC50 = 480 nM T75243 C84TLP 44606820 IC50 = 170 nM T75243 C3H4EB 44606823 IC50 = 27 nM T75243 CD4A8G 44606998 IC50 = 111 nM T75243 C80RQK 44606999 IC50 = 73 nM T75243 CFW9G3 44607000 IC50 = 9.6 nM T75243 CHL59X 44607001 IC50 = 113 nM T75243 C7H3RM 44607002 IC50 = 145 nM T75243 C2TJ3K 44607003 IC50 = 16 nM T75243 CHM5T4 44607180 IC50 = 20 nM T75243 C85XWN 44607181 IC50 = 200 nM T75243 C52ILQ 44607183 IC50 = 12 nM T75243 C2UP6C 44607528 IC50 = 76 nM T75243 CH6OY3 44607529 IC50 = 84 nM T75243 CH6V9F 44608754 IC50 = 3.9 nM T75243 C0IY9N 44608757 IC50 = 5.3 nM T75243 C90ITS 44608915 IC50 = 3.9 nM T75243 CZH1P9 44609387 IC50 = 5 nM T75243 CNDX48 44609388 IC50 = 37 nM T75243 C4TS8G 44610775 IC50 = 21 nM T75243 CAE82W 44623107 IC50 < 1 nM T75243 CYGA93 44814560 Ki = 12 nM T75243 CV24XP 44814563 Ki = 6.6 nM T75243 C37AQP 44815590 Ki = 9.6 nM T75243 CQVB69 44816122 Ki = 17 nM T75243 CT2Y5W 44816299 Ki = 122 nM T75243 C27ZIX 44816464 Ki = 5.1 nM T75243 C6GA8J 44816634 Ki = 1500 nM T75243 CIS31K 44817154 Ki = 21 nM T75243 C54IUP 44818842 IC50 = 250 nM T75243 C16IMZ 44819024 IC50 = 2.95 nM T75243 CN38JF 44819199 IC50 = 0.57 nM T75243 CVW6L8 44819200 IC50 = 3.7 nM T75243 CZ7M6D 44819201 IC50 = 0.39 nM T75243 C7MU8J 44819203 IC50 = 0.75 nM T75243 C8FU0W 44819375 IC50 = 1.21 nM T75243 C4N8CK 44819376 IC50 = 1.1 nM T75243 C0U1IR 45139233 Ki = 500 nM T75243 CK49WN 45139234 Ki = 3900 nM T75243 CYP0M7 45254032 IC50 = 5.4 nM T75243 C1BRW8 45254590 Ki = 4.51 nM T75243 CQ92ME 45379087 Ki = 396 nM T75243 C5I1VH 45379222 IC50 = 11.3 nM T75243 CA4JZ8 45379223 IC50 = 2.3 nM T75243 C12QFV 45480167 Ki = 840 nM T75243 C4V5DT 45482916 IC50 = 0.62 nM T75243 CAL96M 45482923 IC50 = 0.16 nM T75243 C8T6ML 45482926 IC50 = 0.22 nM T75243 C5C2YW 45482931 IC50 = 84 nM T75243 CP45HK 45482935 IC50 = 0.17 nM T75243 CR93VD 45482947 IC50 = 0.2 nM T75243 CDXB49 45482952 IC50 = 0.56 nM T75243 CCS97L 45482982 IC50 = 0.2 nM T75243 CX4TC8 45483330 IC50 = 575 nM T75243 C28OEC 45487702 IC50 = 1500 nM T75243 C38HVQ 45487703 IC50 = 5500 nM T75243 COXA34 45487715 IC50 = 510 nM T75243 C36DZY 45487716 IC50 = 520 nM T75243 CJ7U6H 45487737 IC50 > 10000 nM T75243 CNHR02 45487749 IC50 = 570 nM T75243 CV81ML 45487755 IC50 = 180 nM T75243 CF3TV5 45488020 IC50 = 13 nM T75243 CPLM59 45488021 IC50 = 51 nM T75243 CIL9W1 45488031 IC50 = 1.1 nM T75243 C2Q9ID 45488032 IC50 = 0.2 nM T75243 CA98FY 45488033 IC50 = 0.7 nM T75243 CH07NQ 45488034 IC50 = 0.8 nM T75243 CB8DE0 45488052 IC50 = 0.1 nM T75243 CF3LV9 45488056 IC50 = 2.7 nM T75243 CCL46I 45488057 IC50 = 0.7 nM T75243 CP58QK 45488058 IC50 = 0.1 nM T75243 C9S4MU 45488059 IC50 = 0.3 nM T75243 C0V7UL 45488060 IC50 = 0.2 nM T75243 C8YEC5 45488061 IC50 = 0.2 nM T75243 C6RTH4 45488066 IC50 = 0.9 nM T75243 CWN8V6 45488069 IC50 = 1.5 nM T75243 C1YM6P 45488070 IC50 = 0.3 nM T75243 CNK52A 45488071 IC50 = 1 nM T75243 CO8T6V 45488077 IC50 = 0.3 nM T75243 CBAT68 45488078 IC50 = 6 nM T75243 CZ68MG 45488079 IC50 = 0.6 nM T75243 CFOH35 45488080 IC50 = 0.2 nM T75243 CE3Q7D 45488081 IC50 = 1.7 nM T75243 CI3FZ2 45488082 IC50 = 0.9 nM T75243 CV1U7I 46180604 Ki = 29 nM T75243 CZGB46 46180666 IC50 = 750 nM T75243 CASO36 46182743 Ki = 6.8 nM T75243 C4HFV9 46190734 IC50 = 1.8 nM T75243 CTZD58 46190735 IC50 = 1.1 nM T75243 C61ZLI 46190736 IC50 > 4000 nM T75243 C0V5FS 46190794 IC50 = 66 nM T75243 CA36SV 46191509 IC50 = 336 nM T75243 C5V1DM 46191571 IC50 = 287 nM T75243 CV89YR 46191573 IC50 = 396 nM T75243 C2VJQ1 46191628 IC50 = 230 nM T75243 CR9SZ1 46191757 IC50 = 66.5 nM T75243 CP8DY9 46191758 IC50 = 45.9 nM T75243 C6H3GT 46196486 IC50 = 0.8 nM T75243 CL08DK 46201895 IC50 = 1.4 nM T75243 CL4U2V 46202650 Ki = 110 nM T75243 CX3D9U 46202651 Ki = 106 nM T75243 C9PC6U 46202652 Ki = 203 nM T75243 CHDX80 46202976 IC50 = 729 nM T75243 CI47RP 46206016 IC50 = 23 nM T75243 C3Z6BX 46206784 IC50 = 1 nM T75243 C1D4TK 46214389 IC50 = 90 nM T75243 C1RNM6 46214392 IC50 = 122 nM T75243 C93ZNA 46215208 IC50 = 68 nM T75243 CX8S2G 46215210 IC50 = 18 nM T75243 CF57GK 46215462 IC50 > 10000 nM T75243 CGMS50 46215563 IC50 = 90 nM T75243 CRBF57 46215564 IC50 = 108 nM T75243 CO1D6B 46215565 IC50 = 149 nM T75243 CDA3R9 46220225 Ki > 10000 nM T75243 CIJ5V9 46224766 IC50 = 720 nM T75243 CIPV59 46224808 IC50 = 2050 nM T75243 C4SQY2 46225156 IC50 = 3.3 nM T75243 CL89JZ 46225157 IC50 = 2.5 nM T75243 CFB7Y4 46225158 IC50 = 7.2 nM T75243 C65IPQ 46225280 IC50 = 870 nM T75243 C8A7QJ 46225281 IC50 = 200 nM T75243 CPL45H 46225307 IC50 = 8900 nM T75243 CU12LG 46227561 IC50 = 35 nM T75243 CU0T1P 46227563 IC50 = 100 nM T75243 CK20PN 46227564 IC50 = 22 nM T75243 C3VB6I 46227571 IC50 = 26.5 nM T75243 CS03RK 46227572 IC50 = 0.29 nM T75243 CO4J6R 46227578 IC50 = 11 nM T75243 CO14HC 46227579 IC50 = 0.44 nM T75243 CM1A2S 46227582 IC50 = 20 nM T75243 CT2CH5 46227596 IC50 = 0.9 nM T75243 CG26LH 46227597 IC50 = 1.4 nM T75243 CXW1N8 46227599 IC50 = 0.7 nM T75243 CO64ZL 46227600 IC50 = 0.7 nM T75243 CBF0O4 46227603 IC50 = 16 nM T75243 C2Z4WI 46227604 IC50 = 1 nM T75243 C76PKV 46227605 IC50 = 4.7 nM T75243 C3JK1T 46227606 IC50 = 0.6 nM T75243 CV9O8I 46227607 IC50 = 3.7 nM T75243 CW25EH 46227608 IC50 = 0.45 nM T75243 C5FU9E 46227614 IC50 = 58 nM T75243 C59UJH 46227615 IC50 = 0.34 nM T75243 CS3A9G 46227620 IC50 = 0.68 nM T75243 CG29EB 46227625 IC50 = 1.25 nM T75243 CI9CJ1 46227632 IC50 = 57 nM T75243 CL34IK 46227801 IC50 = 290 nM T75243 C6D2RL 46227820 IC50 = 90 nM T75243 CSIK15 46228569 IC50 = 460 nM T75243 C18WPC 46232643 IC50 = 0.12 nM T75243 CF4WB3 46232644 IC50 = 2.85 nM T75243 C7LKA5 46232645 IC50 = 14.5 nM T75243 C3ZP0G 46232682 IC50 = 0.33 nM T75243 CLE2O9 46232721 IC50 = 0.74 nM T75243 C4IA5M 46232759 IC50 = 1.19 nM T75243 C64HAE 46232760 IC50 = 0.26 nM T75243 CIMH64 46232761 IC50 = 0.22 nM T75243 C47ZSV 46232801 IC50 = 0.22 nM T75243 CVF7G6 46232802 IC50 = 0.16 nM T75243 CXP84Y 46232803 IC50 = 0.12 nM T75243 CT2O8D 46232804 IC50 = 0.12 nM T75243 CL7C2K 46244173 IC50 = 180 nM T75243 C2NH0A 46244259 IC50 = 230 nM T75243 CVJM38 46244260 IC50 = 3300 nM T75243 C79JGP 46830152 IC50 = 5.4 nM T75243 CC62SY 46830153 IC50 = 9 nM T75243 CU4T7F 46830277 IC50 = 3.1 nM T75243 CZ3WS1 46861592 IC50 = 0.2 nM T75243 C7H4YM 46865419 IC50 > 10000 nM T75243 CRO8W0 46865423 IC50 = 3 nM T75243 C47VTS 46865424 IC50 = 10 nM T75243 C7Q4OP 46865531 Ki = 5 nM T75243 C7T4RN 46865885 IC50 = 1 nM T75243 CO3P0J 46866604 IC50 = 0.46 nM T75243 CQ2Y1V 46866705 Ki = 1.42 nM T75243 C62NFQ 46883920 IC50 = 5.6 nM T75243 CKJ2D4 46883989 IC50 = 57 nM T75243 C82RWD 46883990 IC50 = 3500 nM T75243 CE3B7R 46883991 IC50 = 3.45 nM T75243 CP9JO4 46884017 IC50 = 145 nM T75243 C18KOY 46884018 IC50 = 14.3 nM T75243 C9RD8J 46884019 IC50 = 29 nM T75243 CP3C4Z 46884064 IC50 = 71 nM T75243 C65AQI 46884065 IC50 = 10.5 nM T75243 C7NK1H 46884066 IC50 = 115 nM T75243 C3BV5E 46884067 IC50 = 18 nM T75243 C9LB7I 46884068 IC50 = 17 nM T75243 CLOR10 46884069 IC50 = 70 nM T75243 CE70MJ 46884070 IC50 = 8.2 nM T75243 CIAK59 46884071 IC50 = 47.5 nM T75243 CO09QJ 46884072 IC50 = 8.2 nM T75243 CK95YV 46884073 IC50 = 10.9 nM T75243 CUI09D 46884074 IC50 = 9.3 nM T75243 CUL4I2 46884075 IC50 = 8.4 nM T75243 C9MHF4 46884076 IC50 = 102.5 nM T75243 CHM48L 46884077 IC50 = 13 nM T75243 C6MZ1J 46884121 IC50 = 800 nM T75243 C96FTP 46884122 IC50 = 33 nM T75243 C5RM6X 46884123 IC50 = 42 nM T75243 CKT35D 46884156 IC50 = 19 nM T75243 CFP9B5 46884157 IC50 = 0.55 nM T75243 CI3U2Q 46884158 IC50 = 0.5 nM T75243 CTVN70 46884203 IC50 = 0.56 nM T75243 C4FC9H 46884204 IC50 = 2 nM T75243 CEJ9C3 46884242 IC50 = 1 nM T75243 C8S5TR 46884243 IC50 = 0.39 nM T75243 CU93BN 46884282 IC50 = 1.85 nM T75243 C2H5CE 46884283 IC50 = 4.55 nM T75243 CWFH78 46884284 IC50 = 18 nM T75243 CZ5M8O 46884285 IC50 = 180 nM T75243 CV3C0K 46884353 IC50 = 0.72 nM T75243 CZV8T9 46884354 IC50 = 17 nM T75243 CO9W8A 46884355 IC50 = 19 nM T75243 CLA01F 46884356 IC50 = 2.2 nM T75243 CO1D2H 46884404 IC50 = 0.38 nM T75243 CB6YM8 46884405 IC50 = 2.1 nM T75243 CL8PR5 46884406 IC50 = 2.75 nM T75243 CY9M0N 46884525 IC50 = 0.18 nM T75243 CH0QN3 46884526 IC50 = 0.7 nM T75243 CAU6E8 46884527 IC50 = 5.4 nM T75243 CA2U0D 46884528 IC50 = 6.6 nM T75243 C5JBC1 46884529 IC50 = 8.8 nM T75243 CH2RD9 46884530 IC50 = 1.2 nM T75243 CWHK39 46884531 IC50 = 0.7 nM T75243 CSQ5I3 46884532 IC50 = 0.52 nM T75243 CS0Q3T 46884533 IC50 = 0.535 nM T75243 CO5H2J 46884534 IC50 = 0.56 nM T75243 C31KXQ 46884535 IC50 = 0.88 nM T75243 C86PXB 46884536 IC50 = 0.56 nM T75243 C6TI7E 46884537 IC50 = 0.81 nM T75243 CRW39C 46884538 IC50 = 0.34 nM T75243 C02IJK 46884539 IC50 = 0.14 nM T75243 C4SX6O 46884540 IC50 = 0.7 nM T75243 CE5S7W 46884541 IC50 = 0.4 nM T75243 CAS1R6 46884542 IC50 = 1.2 nM T75243 C87UVQ 46884543 IC50 = 1.25 nM T75243 C2RJ4E 46884544 IC50 = 0.9 nM T75243 CE8YC5 46884545 IC50 = 0.42 nM T75243 CM3C9U 46884546 IC50 = 0.1 nM T75243 CGY1E3 46884547 IC50 = 1.7 nM T75243 CUPR76 46885272 IC50 = 0.25 nM T75243 CHP18Q 46885273 IC50 = 0.57 nM T75243 CY89OZ 46885274 IC50 = 0.57 nM T75243 CZ1XR9 46885275 IC50 = 1 nM T75243 C9N5RS 46885276 IC50 = 1.1 nM T75243 CZYO07 46885277 IC50 = 0.89 nM T75243 C1Y7QN 46885278 IC50 = 1.6 nM T75243 CNLX49 46885279 IC50 = 0.9 nM T75243 CSA92E 46885280 IC50 = 0.8 nM T75243 CL4ZI9 46885281 IC50 = 0.26 nM T75243 CN3RH4 46885425 IC50 = 9200 nM T75243 CLA40T 46885426 IC50 = 11000 nM T75243 COL95X 46885494 IC50 = 5000 nM T75243 CVWU94 46885495 IC50 = 500 nM T75243 CC8T1E 46885496 IC50 = 190 nM T75243 CM8JX9 46885534 IC50 = 22 nM T75243 CCS20H 46885565 IC50 = 1 nM T75243 CG47YP 46885566 IC50 = 62 nM T75243 C4R3XP 46885599 IC50 = 4 nM T75243 C3SMV1 46885600 IC50 = 96 nM T75243 CV5MK6 46885601 IC50 = 215 nM T75243 C2M1DN 46885624 IC50 = 108 nM T75243 C42WVO 46885648 IC50 = 7 nM T75243 C0ZV8M 46886360 Ki = 10 nM T75243 C1JS5T 46886361 Ki = 50 nM T75243 CGRO36 46886375 Ki = 4 nM T75243 CZR3V2 46886410 Ki = 4 nM T75243 C4PRU3 46891423 IC50 = 1.3 nM T75243 CXPZ24 46891467 IC50 = 5.2 nM T75243 C9G4IW 46891468 IC50 = 2.4 nM T75243 C4IW0N 46891469 IC50 = 1.5 nM T75243 CF17MQ 46891470 IC50 = 4.2 nM T75243 CRHK80 46891471 IC50 = 3.8 nM T75243 C9SUH8 46891472 IC50 = 1.1 nM T75243 CGME41 46891473 IC50 = 2.5 nM T75243 C3HMQ2 46891474 IC50 = 0.3 nM T75243 CARY94 46891475 IC50 > 4000 nM T75243 CP38DV 46891889 Ki = 9 nM T75243 CB6Z8P 46892208 IC50 = 1300 nM T75243 CZX46Y 46892342 IC50 = 1500 nM T75243 C5FN6I 46892845 IC50 = 390 nM T75243 CQ32BN 46892970 IC50 = 150 nM T75243 COJA32 46892971 IC50 = 8 nM T75243 C5QFB3 46893088 IC50 = 27 nM T75243 C1Q8HJ 46893484 IC50 = 370 nM T75243 CO5ZE0 46893618 IC50 = 43 nM T75243 CS30AI 46893754 IC50 = 31 nM T75243 C8ESU7 46912801 Ki = 10 nM T75243 C3HG6N 46913071 Ki = 140 nM T75243 CDGN94 46913265 Ki = 12 nM T75243 CIM9S2 46913471 Ki = 12 nM T75243 CPO1N7 46927938 Ki = 4880 nM T75243 CFO9X3 46946049 IC50 = 989 nM T75243 CL84AF 46946248 IC50 > 10000 nM T75243 CF14PE 46947264 IC50 = 0.42 nM T75243 CMRT49 49780177 IC50 = 966 nM T75243 C2Y9OC 49780178 IC50 = 3810 nM T75243 C4T2GU 49780179 IC50 = 13.5 nM T75243 CLW50G 49780380 IC50 = 78.9 nM T75243 CP92MJ 49780381 IC50 = 93.8 nM T75243 C1TIH2 49780382 IC50 = 3440 nM T75243 C64MFW 49780383 IC50 = 33.2 nM T75243 CL1W9U 49780384 IC50 = 662 nM T75243 CV0I7K 49780592 IC50 = 213 nM T75243 CZ2T5F 49780593 IC50 = 82.6 nM T75243 CKMO53 49780594 IC50 = 214 nM T75243 C3WAJ9 49780595 IC50 = 25.8 nM T75243 CQB86T 49780596 IC50 = 239 nM T75243 CA1IQ0 49780810 IC50 = 95 nM T75243 C0N6SF 49780811 IC50 = 6.84 nM T75243 C5RBK7 49780812 IC50 = 3.6 nM T75243 CG82WE 49780813 IC50 = 0.57 nM T75243 C7AY6O 49781041 IC50 = 389 nM T75243 C91BTF 49781042 IC50 = 1.26 nM T75243 C6QV0A 49781043 IC50 = 21.4 nM T75243 CGU7Y0 49781044 IC50 = 4.25 nM T75243 C74ZTC 49781256 IC50 = 26.6 nM T75243 CC05VI 49781257 IC50 = 51.9 nM T75243 CHX76J 49784892 IC50 = 7800 nM T75243 CA1H8S 49784893 IC50 > 10000 nM T75243 CP2QD0 49784894 IC50 = 4800 nM T75243 CTZG05 49784988 IC50 = 7200 nM T75243 CE9AC5 49785078 IC50 = 560 nM T75243 CG2IO7 49785079 IC50 = 530 nM T75243 C8EYN4 49785083 IC50 > 10000 nM T75243 CBNZ47 49785166 IC50 > 10000 nM T75243 CZI34V 49785167 IC50 > 10000 nM T75243 CJK65T 49785253 IC50 = 360 nM T75243 CXK8F5 49785436 IC50 > 10000 nM T75243 CWL5C6 49785518 IC50 > 10000 nM T75243 C3NV0J 49785827 IC50 = 200 nM T75243 C0OZM2 49785828 IC50 > 10000 nM T75243 C1AR4G 49785829 IC50 > 10000 nM T75243 C39HAK 49785832 IC50 > 10000 nM T75243 CA53NO 49788443 IC50 = 237 nM T75243 C9K1XO 49800133 Ki = 0.85 nM T75243 C3D2RG 49800134 Ki = 5.11 nM T75243 CQ93PT 49800135 Ki = 5 nM T75243 CWI3E0 49800136 Ki = 0.8 nM T75243 C9ZW3R 49835055 IC50 = 12 nM T75243 CI6B7G 49835106 IC50 = 37 nM T75243 CN2E0P 49835107 IC50 = 13 nM T75243 CV50DY 49835108 IC50 = 198 nM T75243 CTM6U1 49835172 IC50 = 121 nM T75243 CL6V8Y 49835227 IC50 = 35 nM T75243 C90XTJ 49835286 IC50 = 3 nM T75243 CA4NH7 49850583 IC50 = 5000 nM T75243 CT4Y6E 49852123 IC50 > 50000 nM T75243 CXOH76 49855456 Ki = 3.2 nM T75243 C08PSJ 49855457 Ki = 3.6 nM T75243 CFHP43 49855648 Ki = 1.7 nM T75243 CEPR84 49856040 Ki = 1.3 nM T75243 CP2LC8 49857180 Ki = 10 nM T75243 CWT1P9 49857571 Ki = 1.4 nM T75243 CJ21VU 49857572 Ki = 4.4 nM T75243 C5E0JI 49858150 Ki = 0.7 nM T75243 C6JBA1 49858345 Ki = 3 nM T75243 C1C2UI 49858346 Ki = 1.6 nM T75243 CY8MP7 49867926 IC50 = 190 nM T75243 C25YNT 50940492 Ki = 5 nM T75243 C2Q0GE 50990922 IC50 = 93 nM T75243 CKY3V1 50990924 IC50 = 2 nM T75243 CGQ49I 51003483 Ki = 3 nM T75243 C0HWJ7 51003484 Ki = 13 nM T75243 CHP3Z4 51003485 Ki = 265 nM T75243 CPA8N1 51039139 Ki = 8 nM T75243 CLZ8N6 51352027 IC50 = 6.31 nM T75243 C73ANH 51353707 IC50 = 57 nM T75243 CI4A6R 51353708 IC50 = 285 nM T75243 CJ4ZL6 51353709 IC50 = 262 nM T75243 CDLF71 51353710 IC50 = 45 nM T75243 C04EVK 51353711 IC50 > 6000 nM T75243 CD6AL8 51353712 IC50 = 47 nM T75243 CPQ1G6 51354021 IC50 = 719 nM T75243 CVK95R 51354022 IC50 = 65 nM T75243 CHKA96 51354023 IC50 = 269 nM T75243 CRL1B8 51354025 IC50 > 6000 nM T75243 C6VD0B 51354313 IC50 = 29 nM T75243 CJC90Y 51354315 IC50 = 11 nM T75243 COH9L7 51354317 IC50 = 15 nM T75243 CV6I5D 51354595 IC50 = 1500 nM T75243 C1V6RN 51354597 IC50 = 1.6 nM T75243 CZ32XV 51354599 IC50 = 6 nM T75243 C8WEN4 51354600 IC50 = 2.1 nM T75243 C76KOV 51354878 IC50 < 1 nM T75243 CA3O2L 51354879 IC50 < 1 nM T75243 C0O2PW 51354880 IC50 = 1.6 nM T75243 C3JV4L 51354881 IC50 < 1 nM T75243 C6NL1Z 51354882 IC50 < 1 nM T75243 CPWD73 51354883 IC50 < 1 nM T75243 C9CYA1 51355056 Ki = 150 nM T75243 C6E9WP 51355057 Ki = 30 nM T75243 C4QE1V 51355058 Ki = 69 nM T75243 CB10AP 51355171 IC50 = 2.1 nM T75243 CKE42Q 51355172 IC50 = 2.1 nM T75243 CZF89J 51355173 IC50 = 1.1 nM T75243 CQF0J9 51355174 IC50 = 2.3 nM T75243 CO7M9F 51355343 Ki = 4 nM T75243 CJ0KM6 51355344 Ki = 120 nM T75243 CT0V8F 51355345 Ki = 40 nM T75243 C0R8XN 51355348 Ki = 2 nM T75243 C7KT4Z 51355620 Ki = 1 nM T75243 CI71WE 51355621 Ki = 28 nM T75243 CLH35Z 51355622 Ki = 30 nM T75243 C2ODW5 51357942 IC50 > 6000 nM T75243 CSR12N 51357943 IC50 > 6000 nM T75243 CT8LF4 51357944 IC50 > 6000 nM T75243 C8IOD1 51357945 IC50 > 6000 nM T75243 C1KB9V 51357946 IC50 > 6000 nM T75243 C7HOD9 51357947 IC50 > 6000 nM T75243 CI7MJ6 51357948 IC50 > 6000 nM T75243 CRJ5W8 51358113 IC50 = 0.25 nM T75243 C9NS6B 52933960 IC50 = 41 nM T75243 CM24LF 52938983 IC50 = 3018 nM T75243 CU1P2L 52940797 IC50 = 100000 nM T75243 CD62QJ 52940982 IC50 = 93.5 nM T75243 C43SVQ 52941322 IC50 = 0.8 nM T75243 CK59HM 52941479 IC50 = 0.5 nM T75243 C3EJ9D 52941545 Ki = 947 nM T75243 C3ZOK1 52941683 Ki = 113 nM T75243 CDHJ08 52942235 IC50 = 10000 nM T75243 CHU8L6 52942777 Ki = 18 nM T75243 CFRN73 52942850 IC50 = 1.3 nM T75243 C4D1KT 52942879 IC50 = 3.45 nM T75243 C1XEV2 52943394 IC50 = 3600 nM T75243 C73WTL 52943744 IC50 = 1.1 nM T75243 C6Q1AH 52943745 IC50 = 1.85 nM T75243 CG7I1F 52943917 Ki = 6 nM T75243 CMG20V 52945133 Ki > 4000 nM T75243 CWD27C 52945142 IC50 = 0.73 nM T75243 CJ25NV 52945145 Ki = 3940 nM T75243 CWPC54 52945348 IC50 = 220 nM T75243 CXL53B 52945589 IC50 = 1.9 nM T75243 C4NLX7 52945630 IC50 = 2400 nM T75243 CXD6T8 52945845 IC50 = 16000 nM T75243 CN8F0V 52946289 IC50 = 13.5 nM T75243 CMQY93 52946368 IC50 = 1.55 nM T75243 C54LRW 52947235 IC50 = 1700 nM T75243 C5X9VO 52948007 IC50 = 3.3 nM T75243 CW9Z1T 52949347 IC50 = 2 nM T75243 CB0KM5 52949869 IC50 = 0.43 nM T75243 CE63PX 52949940 Ki = 5 nM T75243 CAJQ03 52950001 IC50 = 1.26 nM T75243 C5HQ2E 52950102 IC50 = 0.32 nM T75243 C4TNK8 52951283 IC50 = 1800 nM T75243 CJM04D 52951389 IC50 = 2500 nM T75243 C1VOS0 52951390 IC50 = 2100 nM T75243 CE05DT 53236130 Ki = 3 nM T75243 CP0L3O 53236131 Ki = 25 nM T75243 CD9WT7 53236132 Ki = 6 nM T75243 CG5BU3 53236606 Ki = 1.2 nM T75243 C6M0EG 53236607 Ki = 2.6 nM T75243 CFT4D9 53236823 Ki = 0.8 nM T75243 C5IFP3 53236824 Ki = 1.2 nM T75243 CDKV61 53237046 Ki = 1 nM T75243 CAL64M 53237047 Ki = 1.3 nM T75243 CJZ7I0 53237048 Ki = 0.34 nM T75243 C7QGN3 53237049 Ki = 0.66 nM T75243 CAS87Q 53237257 Ki = 4 nM T75243 C23VLY 53237258 Ki = 2.9 nM T75243 C6F5MH 53237259 Ki = 1 nM T75243 CR93EL 53237260 Ki = 1.1 nM T75243 COD8S4 53237261 Ki = 7 nM T75243 C6A3FN 53237262 Ki = 62 nM T75243 CYP5A7 53237477 Ki = 7.9 nM T75243 CIWE59 53237478 Ki = 1.7 nM T75243 CTM6D8 53237479 Ki = 6.8 nM T75243 C3Y8JZ 53237480 Ki = 21 nM T75243 CZ0LW2 53237719 Ki = 2.3 nM T75243 C34ZJA 53237720 Ki = 1.8 nM T75243 C39NBH 53237721 Ki = 3.2 nM T75243 CA85MY 53237722 Ki = 4.7 nM T75243 CT8IN1 53242225 IC50 = 600 nM T75243 C9NF0C 53302364 Ki = 8170 nM T75243 C4J9WZ 53307606 IC50 = 530 nM T75243 C7ZH0D 53308041 IC50 = 3.01 nM T75243 CT54XZ 53316658 Ki = 21 nM T75243 CG6O0M 53317018 Ki = 1330 nM T75243 C8FPQ4 53318293 Ki = 1000 nM T75243 CK9SE2 53318295 Ki = 84 nM T75243 CY8DH9 53322283 Ki = 1000 nM T75243 CN92LK 53322732 IC50 = 4000 nM T75243 CCSP27 53323641 Ki = 31 nM T75243 CW9F1T 53323642 Ki = 162 nM T75243 CQX59J 53323643 Ki = 216 nM T75243 CTD8A0 53324021 Ki = 3250 nM T75243 CZ41DR 53324923 Ki = 984 nM T75243 CZQ80X 53326214 Ki = 66 nM T75243 C25LHM 53326216 Ki = 17 nM T75243 CRYW35 53350231 Ki = 10 nM T75243 CCX7M5 53353847 Ki = 1260 nM T75243 C23HAU 53361718 IC50 = 1.6 nM T75243 CM60WQ 53361719 IC50 = 0.41 nM T75243 CBPR36 53363353 IC50 = 33 nM T75243 CL69DK 53377727 IC50 = 59 nM T75243 CG3C1J 53379513 IC50 = 0.7 nM T75243 C5SMC3 53387410 IC50 = 49 nM T75243 C5Q0HA 53387411 IC50 = 229 nM T75243 C90KZU 53387571 IC50 = 430 nM T75243 CMO9K1 53387572 IC50 = 446 nM T75243 CI40BG 53387573 IC50 = 70 nM T75243 C2IJR7 53387574 IC50 = 76 nM T75243 CWB79U 53387575 IC50 > 25000 nM T75243 CB4H9G 53387738 IC50 = 146 nM T75243 C5ZY9R 53387740 IC50 = 292 nM T75243 CVG90B 53389651 IC50 > 10000 nM T75243 CSV9X2 54579940 IC50 = 2 nM T75243 CN51TL 54579941 IC50 = 270 nM T75243 C7VZU2 54579942 IC50 = 260 nM T75243 C4R9JB 54579943 IC50 = 180 nM T75243 CG26HQ 54579944 IC50 = 80 nM T75243 CQE1Z7 54580062 IC50 = 390 nM T75243 C5O9WP 54580063 IC50 = 2100 nM T75243 CC5R3O 54580924 IC50 = 140 nM T75243 C3OIY4 54580925 IC50 = 45 nM T75243 CUP7N6 54581023 IC50 = 870 nM T75243 CAB63J 54581048 IC50 = 3000 nM T75243 C60TYL 54581049 IC50 = 190 nM T75243 CF2UH5 54581983 IC50 = 180 nM T75243 CB3OM9 54582056 IC50 = 3200 nM T75243 C5B4MV 54582091 IC50 = 110 nM T75243 C23EVN 54582916 IC50 = 680 nM T75243 CI8US3 54582917 IC50 = 33100 nM T75243 CT2SV7 54583916 IC50 = 175 nM T75243 CY87EC 54583917 IC50 = 680 nM T75243 C2GE8J 54584039 IC50 = 2400 nM T75243 C8CPI4 54584859 IC50 = 340 nM T75243 C9TZ2V 54584860 IC50 = 540 nM T75243 CVY42B 54584949 IC50 = 180 nM T75243 C1M9JE 54584986 IC50 = 1900 nM T75243 CME81Q 54585830 IC50 = 250 nM T75243 C81YUR 54585940 IC50 = 34 nM T75243 C1G0IY 54586917 IC50 = 4700 nM T75243 C0Y9ZG 54761473 IC50 = 150 nM T75243 CFUT05 56648675 Ki = 12 nM T75243 C1GAB6 56648677 Ki = 6.3 nM T75243 CWDF40 56648757 Ki = 14 nM T75243 CJO39U 56648759 Ki = 14 nM T75243 C83QGP 56660108 IC50 = 3 nM T75243 CYM1D0 56660109 IC50 = 0.3 nM T75243 CHA35L 56663573 IC50 = 18.5 nM T75243 CF7PY5 56667023 IC50 = 7.7 nM T75243 CC1DJ8 56670464 IC50 = 8.2 nM T75243 CZH95G 56673952 IC50 = 0.4 nM T75243 CHR8K0 56677282 IC50 = 5.6 nM T75243 C79AMB 56677283 IC50 = 22.5 nM T75243 C5ZN6X 56682067 IC50 = 24 nM T75243 CG17TZ 56683916 IC50 = 14.5 nM T75243 C7B2OH 56683917 IC50 = 1.1 nM T75243 C6LMP8 56683918 IC50 = 1.7 nM T75243 C94JIT 56832510 IC50 > 4300 nM T75243 C4Z0OC 56834890 Ki = 2800 nM T75243 C67TJQ 56834891 Ki = 2600 nM T75243 C32CID 56926598 Ki = 3900 nM T75243 CV8Z5C 56926697 Ki = 3900 nM T75243 CO43FQ 56926699 Ki = 1100 nM T75243 C4GT2U 56926701 Ki = 2100 nM T75243 CPGC81 56947516 IC50 > 10000 nM T75243 C0M3EQ 56950791 IC50 = 84 nM T75243 CAK91L 56955954 IC50 = 623 nM T75243 C74YNV 56966983 IC50 = 751 nM T75243 CVK5A3 57328247 IC50 > 10000 nM T75243 CZ7RE0 57345686 IC50 = 32000 nM T75243 C3CL8H 57384862 Ki = 1200 nM T75243 C96WSJ 57387650 Ki = 13 nM T75243 C6I8SF 57390697 IC50 = 3500 nM T75243 C3R2LD 57390793 IC50 = 1590 nM T75243 C9RB7K 57391333 IC50 > 10000 nM T75243 CH37SE 57391335 IC50 > 10000 nM T75243 C0QF7X 57392605 IC50 = 9 nM T75243 C8U6ZC 57392648 IC50 = 120 nM T75243 C7XS2P 57394206 IC50 = 30 nM T75243 CFG53Z 57394325 IC50 > 10000 nM T75243 CSRG42 57394326 IC50 = 2020 nM T75243 C45NDO 57394361 IC50 = 8300 nM T75243 C09MPI 57396034 IC50 = 170 nM T75243 CA52UR 57396083 IC50 = 8900 nM T75243 CS14ZH 57396608 IC50 > 10000 nM T75243 CLJ5B1 57397772 IC50 = 2 nM T75243 C4N7MX 57397773 IC50 = 6 nM T75243 C2XZG9 57397841 IC50 = 390 nM T75243 C2VPR0 57397894 IC50 = 30 nM T75243 CU9N1Z 57398248 IC50 = 71 nM T75243 CQO74C 57398382 IC50 > 10000 nM T75243 CV2Z0C 57398383 IC50 > 10000 nM T75243 C9Z6AL 57399433 IC50 = 10 nM T75243 CA3NV0 57399544 IC50 = 9 nM T75243 C7UYA9 57401258 IC50 = 120 nM T75243 CJC26L 57401330 IC50 > 10000 nM T75243 C0LP7R 57401331 IC50 = 70 nM T75243 CRO5Z6 57401846 IC50 > 10000 nM T75243 CWV56Z 57402952 IC50 = 63 nM T75243 C5TPX8 57403086 IC50 = 130 nM T75243 C8Y7VZ 57427751 IC50 = 758.58 nM T75243 CK6TN2 57427752 IC50 = 5.754 nM T75243 CT6XL0 57466811 IC50 > 9100 nM T75243 C59YAC 57495353 IC50 > 9100 nM T75243 CWQ6F2 57523291 IC50 > 10000 nM T75243 CJE19S 57523686 IC50 > 10000 nM T75243 C1EP6I 58024825 IC50 = 2600 nM T75243 CX8SZ7 58118657 IC50 < 31.62 nM T75243 C46AUK 58137055 IC50 = 262 nM T75243 C7ONC3 58137106 IC50 = 330 nM T75243 C6DH9J 58137111 IC50 = 3160 nM T75243 C7VSX2 58137137 IC50 = 601 nM T75243 C84FUI 58137148 IC50 = 1540 nM T75243 C5IMD7 58137170 IC50 = 1380 nM T75243 CRPL37 58137176 IC50 = 285 nM T75243 CV7YP2 58169819 IC50 = 7.943 nM T75243 CJ8TE4 58169820 IC50 = 12.59 nM T75243 CU3WG8 58298312 IC50 = 106 nM T75243 CONJ64 58298326 IC50 = 30 nM T75243 C0W7QE 58298327 IC50 = 19 nM T75243 C7GIQ1 58298333 IC50 = 175 nM T75243 CB9XN5 58298334 IC50 = 66 nM T75243 C7GA2Y 58379501 Ki = 0.243 nM T75243 C0D7NE 58379507 Ki = 0.842 nM T75243 CO5NX4 58379530 Ki = 18.5 nM T75243 CVL1G3 58379533 Ki = 2.64 nM T75243 C2DM7X 58379543 Ki = 2.2 nM T75243 C5YQL3 58379551 Ki = 2.33 nM T75243 CX01MF 58379559 Ki = 4.71 nM T75243 CT9W7U 58379595 Ki = 1.55 nM T75243 CFE09U 58379619 Ki = 2 nM T75243 C31NXY 58379638 Ki = 47.4 nM T75243 CUTJ73 58379663 Ki = 0.377 nM T75243 CZUO79 58441681 IC50 = 0.75 nM T75243 CB2VP8 58507929 Ki = 19.3 nM T75243 CK0O4B 58508043 Ki = 109 nM T75243 C1I4ZO 58508110 Ki = 64.5 nM T75243 CPCG46 58508197 Ki = 224 nM T75243 C85HOT 58508283 Ki = 25.5 nM T75243 C58FIX 58508310 Ki = 609 nM T75243 CBA73C 59239059 Ki = 48 nM T75243 CDM57O 59239077 Ki = 2.4 nM T75243 C0XN3Y 59239089 Ki = 6.5 nM T75243 CQ4HD1 59239114 Ki = 1.5 nM T75243 CY3M0Z 59239164 Ki = 1.7 nM T75243 C18DJR 59239174 Ki = 6.8 nM T75243 CYOW74 59239188 Ki = 20 nM T75243 C42ZDM 59239194 Ki = 2.4 nM T75243 CRKP62 59239206 Ki = 3 nM T75243 CM0AY7 59239207 Ki = 4.2 nM T75243 CG1A8Y 59239249 Ki = 1.3 nM T75243 COEM65 59239271 Ki = 220 nM T75243 CIR81P 59239300 Ki = 0.4 nM T75243 C82YHL 59239336 Ki = 11 nM T75243 C6MQA3 59239348 Ki = 1.4 nM T75243 CN9WD1 59239356 Ki = 2.3 nM T75243 C6ZRI4 59239369 Ki = 5.5 nM T75243 C2BX0H 59239374 Ki = 18 nM T75243 CQ6I7T 59239380 Ki = 130 nM T75243 CP64KI 59239424 Ki = 2.7 nM T75243 CVG8B3 59239456 Ki = 3.5 nM T75243 CTX01P 59239521 Ki = 2.7 nM T75243 C4YW3N 59239622 Ki = 3.7 nM T75243 CDX4G0 59258834 Ki = 51.2 nM T75243 CY0SB7 59258852 Ki = 76.4 nM T75243 CSJ60G 59258855 Ki = 23.5 nM T75243 CSIV71 59258894 Ki = 110 nM T75243 CCZ9F4 59258904 Ki = 700 nM T75243 C36ZSD 59258941 Ki = 10.6 nM T75243 CJ4ME2 59258944 Ki = 190 nM T75243 C4SRU6 59258964 Ki = 18.6 nM T75243 COA89E 59258965 Ki = 82 nM T75243 CUF6Y9 59259010 Ki = 150 nM T75243 CD43UI 59259014 Ki = 272 nM T75243 C3NKS2 59259019 IC50 = 30.09 nM T75243 CI2SU0 59453028 IC50 = 8 nM T75243 CY8L4O 59453029 IC50 = 12 nM T75243 CTMA05 59453047 IC50 = 14 nM T75243 C8YDC3 59453057 IC50 = 103 nM T75243 CYN1L2 59453060 IC50 = 103 nM T75243 CA4XV9 59453066 IC50 = 25 nM T75243 C1I7QA 59453069 IC50 = 5 nM T75243 CNV0I9 59453076 IC50 = 38 nM T75243 CQYI53 59453077 IC50 = 12 nM T75243 CV6A4J 59453078 IC50 = 8 nM T75243 CM2Q5J 59453081 IC50 = 3 nM T75243 CV1SY9 59453083 IC50 = 185 nM T75243 CPH5N4 59453087 IC50 = 436 nM T75243 CRFC53 59453089 IC50 = 15 nM T75243 C1RTQ6 59453093 IC50 = 33 nM T75243 C26QRA 59453105 IC50 = 37 nM T75243 C2BM8E 59453110 IC50 = 26 nM T75243 C0WQ4N 59453111 IC50 = 4 nM T75243 CO9G5I 59453117 IC50 = 72 nM T75243 CWJ3L7 59453121 IC50 = 4 nM T75243 CLQ08G 59453125 IC50 = 168 nM T75243 CXA9D8 59453133 IC50 = 46 nM T75243 C5D6ZW 59477194 IC50 = 385 nM T75243 C2X8TY 59548177 IC50 > 10000 nM T75243 C71GBC 59548184 IC50 > 10000 nM T75243 C10NEZ 59548195 IC50 > 25000 nM T75243 CGRO45 59548196 IC50 > 10000 nM T75243 CD39AG 59548207 IC50 > 10000 nM T75243 C5B0MY 59548213 IC50 = 10600 nM T75243 C6KP4G 59548220 IC50 > 10000 nM T75243 CL82RM 59548221 IC50 > 10000 nM T75243 CTNU85 59548226 IC50 > 10000 nM T75243 CLF4I3 59548231 IC50 = 6700 nM T75243 CLB6N4 59548232 IC50 = 5100 nM T75243 C2KBG8 59548236 IC50 > 10000 nM T75243 CSWV07 59548243 IC50 > 10000 nM T75243 CN48VL 59548245 IC50 > 10000 nM T75243 CMT2R0 59548250 IC50 > 10000 nM T75243 CT5RK1 59548255 IC50 > 16000 nM T75243 C3I8NE 59548256 IC50 > 10000 nM T75243 C8W5HT 59548263 IC50 > 10000 nM T75243 C4WOJ7 59548265 IC50 = 2500 nM T75243 CT8Q5B 59548274 IC50 > 10000 nM T75243 C8FSH7 59548276 IC50 = 2100 nM T75243 CBG52T 59548278 IC50 > 10000 nM T75243 CVF1B2 59548283 IC50 > 10000 nM T75243 CY31EA 59548284 IC50 > 10000 nM T75243 CO4GT7 59548288 IC50 = 163 nM T75243 CFR7S8 59548302 IC50 = 2500 nM T75243 CRE8B3 59548316 IC50 > 10000 nM T75243 C7I9QW 59548318 IC50 = 3700 nM T75243 CRM20Z 59548320 IC50 > 10000 nM T75243 CX1KJ9 59548322 IC50 > 10000 nM T75243 CJE5I4 59548341 IC50 > 10000 nM T75243 CSFV40 59548348 IC50 = 2200 nM T75243 C8O1VS 59548349 IC50 = 3600 nM T75243 CE9W0K 59548355 IC50 > 10000 nM T75243 CWC65A 59548356 IC50 > 10000 nM T75243 CMKP95 59548371 IC50 > 10000 nM T75243 C72TQL 59548376 IC50 > 22000 nM T75243 CC8UV3 59548383 IC50 = 290 nM T75243 CK7ZS8 59548389 IC50 > 17000 nM T75243 C4SN3U 59548390 IC50 > 10000 nM T75243 C5O3BM 59548393 IC50 = 7800 nM T75243 CD4ET2 59548402 IC50 > 10000 nM T75243 CES59T 59548403 IC50 > 10000 nM T75243 CE8P3G 59548407 IC50 = 32 nM T75243 CO4K2W 59548419 IC50 = 74 nM T75243 CSDB78 59548424 IC50 > 10000 nM T75243 C81FCQ 59548431 IC50 > 10000 nM T75243 CLGY34 59548453 IC50 > 10000 nM T75243 CBT21W 59548454 IC50 > 10000 nM T75243 C9DIB3 59548458 IC50 > 10000 nM T75243 CJT68K 59548460 IC50 > 10000 nM T75243 C9LFT3 59548462 IC50 > 10000 nM T75243 C6PVN9 59548463 IC50 = 7800 nM T75243 CA47YQ 59548474 IC50 > 10000 nM T75243 CX8C2U 59548480 IC50 > 10000 nM T75243 CM8PD7 60150509 IC50 = 6300 nM T75243 C5KD3Z 60154714 IC50 > 10000 nM T75243 CS0L4D 60154996 IC50 > 10000 nM T75243 C1UI3P 60155086 IC50 > 10000 nM T75243 CX08ON 60155087 IC50 > 10000 nM T75243 CX8J1I 60155265 IC50 > 10000 nM T75243 CAT40I 60155266 IC50 > 10000 nM T75243 CD56VA 60155268 IC50 = 1400 nM T75243 C5FI4P 60155451 IC50 = 3700 nM T75243 CX9G4U 60155452 IC50 = 1400 nM T75243 CR7EG9 60155538 IC50 > 10000 nM T75243 CU6YB9 60155539 IC50 > 10000 nM T75243 CSZA16 60155724 IC50 = 1781 nM T75243 C6BY2S 60210977 IC50 = 890 nM T75243 C6GE5S 62705166 Ki = 663 nM T75243 C94MTA 62705167 Ki = 123 nM T75243 CV0MD4 62705168 Ki = 13 nM T75243 CSD3F8 62705169 Ki = 15 nM T75243 C3LS8Q 62705170 Ki = 52 nM T75243 C2E3AO 62705171 IC50 = 6 nM T75243 CSD0N6 62705990 IC50 = 15 nM T75243 C9NI6K 62705991 IC50 = 27 nM T75243 C2RDA4 62706154 IC50 = 6 nM T75243 C3M6QC 62706155 IC50 = 3 nM T75243 CAG23H 62706156 IC50 = 3 nM T75243 C1RB8F 62706157 IC50 = 21 nM T75243 CGC62F 62706158 IC50 = 2 nM T75243 C67TAB 62706159 IC50 = 39 nM T75243 C4IGR0 62706312 IC50 = 4 nM T75243 CPM5R9 62706313 IC50 = 2 nM T75243 CX6IU3 62706314 IC50 = 3 nM T75243 CFJ8W5 62706315 IC50 = 10 nM T75243 CX0H7E 62706316 IC50 = 5 nM T75243 C06IUA 62706317 IC50 = 2 nM T75243 C82NPI 62706470 IC50 = 3 nM T75243 CPR50J 62706471 IC50 = 76 nM T75243 CA31ZB 62706472 IC50 = 65 nM T75243 CWRJ86 62706475 IC50 = 63 nM T75243 CNMX21 62706476 IC50 = 141 nM T75243 CS0CA6 62706650 IC50 = 3 nM T75243 C71APZ 62706651 IC50 = 6 nM T75243 CFBD83 62706652 IC50 = 147 nM T75243 CL20FV 62706653 IC50 = 24 nM T75243 C34MPU 62706654 IC50 = 36 nM T75243 CHX01T 62706655 IC50 = 55 nM T75243 CM39TP 62706813 IC50 = 9 nM T75243 CHK4I1 62706814 IC50 = 67 nM T75243 C16ZGX 62706815 IC50 = 15 nM T75243 CS4VA8 62706816 IC50 = 16 nM T75243 CY0D8M 62706817 IC50 = 20 nM T75243 C9G5NA 62707451 Ki = 25 nM T75243 CWZ1I7 62707452 Ki = 50 nM T75243 C7ZY3Q 62707454 Ki = 120 nM T75243 C80KUA 62707599 Ki = 5 nM T75243 C9RV1U 62707603 Ki = 7 nM T75243 CU2P1Z 62707604 Ki = 62 nM T75243 CUC7B3 66557964 IC50 = 42000 nM T75243 CWZ54O 66600540 IC50 > 10000 nM T75243 C6Q0KU 66612050 IC50 > 10000 nM T75243 C0X9FR 66699750 IC50 = 2 nM T75243 CB8WP9 66788776 IC50 = 34 nM T75243 C51ARE 66788835 IC50 = 206 nM T75243 C6DYG9 66788911 IC50 = 412 nM T75243 CQ5TC4 66789238 IC50 = 20 nM T75243 CIR86Z 66789609 IC50 = 57 nM T75243 CYKD92 66789704 IC50 = 36 nM T75243 CRO34N 66790135 IC50 = 157 nM T75243 COE7X1 66790311 IC50 = 12 nM T75243 CUJB72 66790335 IC50 = 62 nM T75243 CU58AM 67073110 Ki = 2470 nM T75243 C1K5PQ 67094257 Ki = 8 nM T75243 CJ46YU 67094333 Ki = 12 nM T75243 CT9AH0 67178880 Ki = 3.2 nM T75243 CIT38E 67179786 Ki = 4.4 nM T75243 CA1WS0 67276196 Ki = 1.4 nM T75243 C4MX9K 67276455 Ki = 4.8 nM T75243 C9LI0M 67294297 Ki = 1700 nM T75243 C1HBC0 67535197 IC50 = 1.7 nM T75243 CNZ2C3 67535447 IC50 = 277 nM T75243 C3M1OJ 67535551 IC50 = 16 nM T75243 C97SXL 68194826 IC50 = 316.23 nM T75243 CJ2BU0 68195106 IC50 > 2000 nM T75243 C3VKM5 68512988 IC50 > 15000 nM T75243 C2D4BQ 68518711 IC50 = 11100 nM T75243 CC63RO 68893189 IC50 = 2 nM T75243 C45TIJ 69489467 IC50 = 1260 nM T75243 CNX20F 70676303 Ki = 9 nM T75243 CM8H3V 70676450 Ki = 21 nM T75243 CDMO03 70682114 IC50 = 2290 nM T75243 C65LPD 70684413 Ki = 50 nM T75243 CG95EC 70684794 IC50 = 5710 nM T75243 CQS8G7 70686830 IC50 > 9100 nM T75243 CMC74I 70688479 IC50 > 5000 nM T75243 CQ04ZJ 70689027 IC50 = 5100 nM T75243 CN45VU 70690535 IC50 > 5000 nM T75243 CC64RD 70692128 IC50 = 22500 nM T75243 C7ASK8 70692129 IC50 = 252 nM T75243 CU3WF2 70693248 IC50 = 10000000 nM T75243 C4P9CL 70693798 Ki = 434 nM T75243 CX2JZ1 70694178 IC50 > 100000 nM T75243 C7HW2B 70694179 IC50 = 37 nM T75243 CICE82 70694721 IC50 > 5000 nM T75243 C38LWS 70694722 IC50 > 5000 nM T75243 CLY5G3 70695401 IC50 > 30000 nM T75243 CF8EK2 71250848 IC50 = 32 nM T75243 CJP69K 71250855 IC50 = 146 nM T75243 C8KD6L 71250859 IC50 = 95 nM T75243 CM10HY 71250872 IC50 = 72 nM T75243 CS3V1R 71250875 IC50 > 500 nM T75243 C85IZO 71250882 IC50 = 48 nM T75243 C1LI6X 71250891 IC50 = 2 nM T75243 CSO29K 71250896 IC50 = 30 nM T75243 CKE7H2 71250907 IC50 = 88 nM T75243 CI5MT1 71250909 IC50 > 500 nM T75243 C9G2MT 71250929 IC50 = 10 nM T75243 CZP1E8 71250935 IC50 = 53 nM T75243 C1MVL0 71273460 Ki = 1840 nM T75243 C6SAW5 71449586 IC50 > 20000 nM T75243 CK58RV 71449587 IC50 = 18 nM T75243 C6GJE3 71451395 IC50 = 4600 nM T75243 CD8Y3S 71451617 IC50 > 10000 nM T75243 C5KH7C 71453205 IC50 = 16 nM T75243 C6VF7J 71453206 IC50 = 18 nM T75243 CR84JX 71453419 IC50 = 7 nM T75243 CZ8Q5P 71454238 IC50 = 198 nM T75243 CO0WF5 71454941 IC50 = 610 nM T75243 CA30GO 71454942 IC50 = 1700 nM T75243 CH3WN6 71454943 IC50 > 4000 nM T75243 CF74SL 71454944 IC50 = 88 nM T75243 CO82IY 71455167 IC50 > 10000 nM T75243 CA7L1Y 71455168 IC50 > 10000 nM T75243 COW5S1 71456726 IC50 = 3300 nM T75243 CZG8I6 71456727 IC50 = 140 nM T75243 CE1IX7 71456728 IC50 = 25 nM T75243 C14OGU 71458568 IC50 = 320 nM T75243 C6CR7L 71458569 IC50 > 20000 nM T75243 CWAU20 71458570 IC50 > 4000 nM T75243 CVQ62G 71458571 IC50 = 110 nM T75243 C74VKX 71458572 IC50 = 3200 nM T75243 CM1ND2 71458573 IC50 = 15 nM T75243 C3S0NP 71458574 IC50 = 45 nM T75243 CY6WI2 71458575 IC50 = 50 nM T75243 C15XAV 71460420 IC50 = 200 nM T75243 CKV1P2 71460421 IC50 = 7.7 nM T75243 CT7K3A 71460422 IC50 = 12 nM T75243 C25FQP 71462104 IC50 > 20000 nM T75243 CY74CX 71472903 IC50 = 16620 nM T75243 CB78IN 71493938 IC50 = 29 nM T75243 CV03AL 71541406 Ki = 13.4 nM T75243 C7V9SQ 71547699 IC50 = 226 nM T75243 CBCW18 71571355 Ki = 8.63 nM T75243 CQ16UM 71584055 IC50 = 190 nM T75243 C1GDL2 71602514 Ki = 12.8 nM T75243 CHV4N8 71602515 Ki = 24.4 nM T75243 C7YVU4 71602573 Ki = 4.46 nM T75243 C90PSW 71602574 Ki = 2.15 nM T75243 C34HNA 71602575 Ki = 19.5 nM T75243 CM06KQ 71602576 Ki = 7.82 nM T75243 COG0X5 71604742 Ki = 4.2 nM T75243 CC5UR3 71604893 Ki = 4.2 nM T75243 COZ4A6 71604894 Ki = 6.5 nM T75243 C13FGZ 71604895 Ki = 14 nM T75243 C4NA0Z 71604896 Ki = 21 nM T75243 CNY35F 71604897 Ki = 2.6 nM T75243 CN08ZO 71605054 Ki = 7.5 nM T75243 CHK8Y6 71605056 Ki = 6.5 nM T75243 C0HEN3 71605057 Ki = 1.2 nM T75243 C2FAE3 71716356 IC50 = 1300 nM T75243 C5K9JV 71717638 Ki = 0.99 nM T75243 C5S8DT 71717639 Ki = 1.2 nM T75243 CJP83B 71719453 Ki = 1.2 nM T75243 C86MQI 71720046 Ki = 1.5 nM T75243 CLT60U 71720047 Ki = 2.1 nM T75243 C7EY1Q 72163951 Ki = 9 nM T75243 CVT76M 72163952 Ki = 7 nM T75243 C9UOH5 72164062 Ki = 6 nM T75243 CT3X8G 72164184 Ki = 19 nM T75243 CLO1P5 72199292 IC50 = 0.6 nM T75243 C9E4XZ 72546233 IC50 > 3000 nM T75243 C29KOU 72709209 IC50 > 10000 nM T75243 CT73IW 72709284 IC50 > 10000 nM T75243 CW6V2I 72947132 IC50 > 2000 nM T75243 CWL0F2 73054768 IC50 = 67 nM T75243 C95YFI 73054769 IC50 = 62 nM T75243 C8EI1X 73673707 IC50 = 3.8 nM T75243 CBYN18 73977439 IC50 = 1622 nM T75243 C9V1YR 73977449 IC50 = 468 nM T75243 CXA90D 73977451 IC50 = 380 nM T75243 CEZ7L2 73977461 IC50 = 1175 nM T75243 CD0T9V 74539799 IC50 = 1.1 nM T75243 C16KOS 74539862 IC50 = 2.2 nM T75243 CKO41J 76310248 IC50 = 100 nM T75243 CEN9Q5 76310249 IC50 = 127 nM T75243 CJCF67 76310250 IC50 = 5 nM T75243 CBI09O 76310352 IC50 = 8.49 nM T75243 CMF0R5 76310353 IC50 = 28.68 nM T75243 C06OME 76310354 IC50 = 62.64 nM T75243 C4BT9H 76314027 IC50 = 125.93 nM T75243 CC8NB4 76314028 IC50 = 18.39 nM T75243 C4MKN3 76317469 IC50 = 1 nM T75243 C3JA4F 76317470 IC50 = 36 nM T75243 C3XYV1 76317571 IC50 = 12.25 nM T75243 CPK6B4 76317572 IC50 = 65.64 nM T75243 C8E4GI 76321204 IC50 = 336 nM T75243 CPLO52 76321296 IC50 = 13.36 nM T75243 CGY1N5 76321297 IC50 > 10000 nM T75243 C34OYK 76321298 IC50 = 35.27 nM T75243 CE35LN 76321299 IC50 = 36.54 nM T75243 CDG8V4 76324821 IC50 = 266 nM T75243 C2BFA1 76324823 IC50 = 400 nM T75243 CZTR31 76324910 IC50 = 35.02 nM T75243 C4FMR8 76324911 IC50 = 13.88 nM T75243 C8X9TV 76324913 IC50 = 11.19 nM T75243 CX3N7R 76328473 IC50 = 2.32 nM T75243 CE5I7T 76328474 IC50 = 39.04 nM T75243 CUC04I 76328475 IC50 = 140.9 nM T75243 C70WJE 76332052 IC50 = 35 nM T75243 CKD7H2 76332159 IC50 > 10000 nM T75243 C8SL3V 76332160 IC50 = 82.12 nM T75243 C3KIG0 76332161 IC50 = 33.92 nM T75243 CZ92PW 76335665 IC50 = 453 nM T75243 C73KJD 76335670 IC50 = 13 nM T75243 CD2KU1 76335780 IC50 = 78.2 nM T75243 C47ZNT 76335781 IC50 = 159.96 nM T75243 CSCK18 76335782 IC50 = 13.91 nM T75243 CRD94L 76335783 IC50 = 171.72 nM T75243 C6VCF1 76335784 IC50 = 8.55 nM T75243 CT1UL6 76335785 IC50 = 19.2 nM T75243 CU86DF 76335786 IC50 = 24.69 nM T75243 C2JTH8 77107528 IC50 > 1000 nM T75243 C42HDP 77107927 IC50 = 580 nM T75243 C04SRC 77147259 IC50 = 1060 nM T75243 C37LKW 86346018 IC50 = 1100 nM T75243 CK8XE9 86652633 IC50 = 328 nM T75243 CNVS32 87343636 Ki = 5410 nM T75243 CB1VI6 90665817 Ki = 16 nM T75243 CP1W6K 91755004 IC50 = 45.8 nM T75243 C64QBH 117995822 Ki = 69 nM T75243 C7KTW4 118000035 Ki = 812 nM T75243 C7E2DY 118000150 Ki = 24 nM T75243 CKZ5N0 118000206 Ki = 1279 nM T75243 C72IRG 118321317 IC50 = 37.6 nM T75243 C7EAJ0 118321318 IC50 = 245 nM T75243 C8AR0W 118321320 IC50 = 79.2 nM T75243 CBE08T 118321322 IC50 = 180 nM T75243 C67XRL 118321324 IC50 = 111 nM T75243 CH7MG0 118321327 IC50 = 67 nM T75243 C1H7SU 118470918 Ki = 284 nM T75243 CM2DO8 118616331 IC50 = 138 nM T75243 CO0YC8 118616775 IC50 = 89.2 nM T75243 C42SYZ 118616923 IC50 = 197.9 nM T75243 CXA8N2 118616927 IC50 = 105.8 nM T75243 C84DGB 118616929 IC50 > 400 nM T75243 C8SRG9 118616951 IC50 = 64 nM T75243 CFQ71C 118616958 IC50 = 108.5 nM T75243 CU6E0P 118616985 IC50 > 400 nM T75243 C7WO2R 118617086 IC50 > 400 nM T75243 CVJU09 118617088 IC50 = 245.7 nM T75243 CQ7A1G 118617093 IC50 = 163.3 nM T75243 C6U0GQ 118617094 IC50 = 153.4 nM T75243 CB5XL3 118617097 IC50 = 223.4 nM T75243 CZ30BK 118617099 IC50 = 119 nM T75243 CGVH36 118617158 IC50 = 66 nM T75243 C4AHL2 118711367 IC50 > 10000 nM T75243 CF5HV8 118720613 IC50 = 1100 nM T75243 C2UIB7 118720614 IC50 > 2300 nM T75243 CSH50J 118720615 IC50 = 4400 nM T75243 C4LW6I 118720885 IC50 > 4600 nM T75243 C9Y4EH 118720886 IC50 = 7500 nM T75243 C9SF2E 118720891 IC50 > 13000 nM T75243 CQV64Y 118722479 IC50 > 15000 nM T75243 CDLC32 118722480 IC50 > 25000 nM T75243 CP9QZ8 118722481 IC50 > 25000 nM T75243 C8Y2AF 118722482 IC50 = 790 nM T75243 C39TEL 118722483 IC50 = 15800 nM T75243 CM4Q5D 118722770 IC50 > 25000 nM T75243 CQCX41 118737057 IC50 > 10000 nM T75243 CKBP72 121231408 IC50 > 10000 nM T75243 CK0LZ1 121275690 IC50 = 1.6 nM T75243 CIN39H 121334370 Ki = 192 nM T75243 CJDS80 121334379 Ki = 12.6 nM T75243 CC1R8L 121334382 Ki = 650 nM T75243 CU37QN 121334400 Ki = 31 nM T75243 CSKB71 121334407 Ki = 73.4 nM T75243 CM2ZS6 121334410 Ki = 60.2 nM T75243 C4R7DN 121334420 Ki = 42.3 nM T75243 CK3G6P 121334425 Ki = 10 nM T75243 C01CNO 121334433 Ki = 7.4 nM T75243 CGCL96 121334436 Ki = 15.3 nM T75243 CB1L6S 121334438 Ki = 42 nM T75243 CV92TK 121334444 Ki = 35 nM T75243 CGD9K5 121334446 Ki = 11.2 nM T75243 CYTA71 121334474 Ki = 3.5 nM T75243 CH6Y9L 121334475 Ki = 13.9 nM T75243 CHX60O 121334481 Ki = 12 nM T75243 CYI09J 121334494 Ki = 13.6 nM T75243 CZ46TQ 121334504 Ki = 10.6 nM T75243 COZT28 121334509 Ki = 6.9 nM T75243 C1YQ8R 121334511 Ki = 32.8 nM T75243 C8M2ET 121334520 Ki = 10.8 nM T75243 C91PVZ 121428416 IC50 = 186 nM T75243 CA2DM0 121428489 IC50 = 2120 nM T75243 CQLX36 121428567 IC50 = 1680 nM T75243 CI1PS7 121428640 IC50 = 13980 nM T75243 C81IFQ 122163152 IC50 = 15 nM T75243 CL36RB 122178108 IC50 = 66.7 nM T75243 C4Q5KS 122178109 IC50 = 3.04 nM T75243 C2BV9G 122178110 IC50 = 0.2 nM T75243 CCHI06 122178111 IC50 = 62.3 nM T75243 C3FS4U 122178112 IC50 = 21.6 nM T75243 CT5J4A 122178113 IC50 = 0.29 nM T75243 C2VGD5 122178120 IC50 = 218 nM T75243 CTE0F7 122178121 IC50 = 363 nM T75243 C3S2UI 122178122 IC50 = 67.9 nM T75243 C57MXE 122178123 IC50 = 345 nM T75243 C24XUZ 122178124 IC50 = 53.6 nM T75243 C3XMW0 122178125 IC50 = 43.7 nM T75243 C2P6KC 122178126 IC50 = 25.8 nM T75243 CS85CU 122181413 IC50 = 15000 nM T75243 CQS67B 122181416 IC50 = 21000 nM T75243 C0NJ3A 122182356 IC50 = 613 nM T75243 CKT74G 122185265 IC50 = 275 nM T75243 CJ6C1O 122185267 IC50 = 123 nM T75243 CD67LU 122705248 IC50 = 8565 nM T75243 CX63VW 122705258 IC50 > 10000 nM T75243 C76IKM 122705261 IC50 = 328 nM T75243 C8ALO2 124088839 IC50 > 10000 nM T75243 C98DKI 127025346 IC50 = 9.9 nM T75243 CBXJ67 127025628 IC50 = 5.4 nM T75243 CB53ZX 127028515 IC50 = 860 nM T75243 CB9VY8 127028516 IC50 = 940 nM T75243 CSV3R7 127029064 IC50 = 78 nM T75243 CAD38Y 127029440 IC50 = 9430 nM T75243 CR17GV 127029715 IC50 = 6260 nM T75243 CQV05N 127032901 IC50 = 114 nM T75243 C0S5WG 127032910 IC50 = 46 nM T75243 CH7QO2 127032911 IC50 = 17 nM T75243 CNA82D 127032912 IC50 > 3000 nM T75243 CMD0Z8 127032913 IC50 > 3000 nM T75243 C59RLZ 127032914 IC50 > 3000 nM T75243 CGKR53 127032915 IC50 = 30 nM T75243 CT3R6Y 127033229 IC50 = 22 nM T75243 CYNX65 127033230 IC50 = 340 nM T75243 CY8UZ1 127033231 IC50 = 310 nM T75243 CKT2Q6 127034306 IC50 = 25 nM T75243 CEF18H 127034307 IC50 = 36 nM T75243 CY1TR5 127035128 IC50 = 1105 nM T75243 CQTE98 127035129 IC50 = 33 nM T75243 CV94GA 127035130 IC50 = 514 nM T75243 CWUK71 127035185 IC50 = 73 nM T75243 C2ZJA9 127035281 IC50 = 30 nM T75243 CW0I4F 127035282 IC50 = 280 nM T75243 CQ3BK8 127035283 IC50 = 674 nM T75243 CJ2E4N 127035335 IC50 = 21 nM T75243 CM9UL5 127035423 IC50 = 51 nM T75243 C7G8JM 127035424 IC50 = 361 nM T75243 CBV03O 127035425 IC50 = 14 nM T75243 CI6D9M 127035790 IC50 = 806 nM T75243 C5ICR3 127035792 IC50 > 3000 nM T75243 C8PO0M 127035794 IC50 = 284 nM T75243 CJK1X6 127035909 IC50 = 24 nM T75243 CZWA79 127035980 IC50 = 1225 nM T75243 C41YQI 127035981 IC50 = 31 nM T75243 CG8DA9 127045861 IC50 = 25 nM T75243 CVF8Z9 127045862 IC50 = 1.8 nM T75243 CH68NT 127046076 IC50 = 5 nM T75243 CA2XD5 127046077 IC50 = 1 nM T75243 C34REM 127046317 IC50 > 50000 nM T75243 CC4ND8 127046862 IC50 = 59 nM T75243 CO25WH 127052538 IC50 > 10000 nM T75243 CK68CA 130453737 IC50 = 21000 nM T75243 CUO41K 130470684 IC50 = 1480 nM T75243 CBY49C 132156028 Ki = 9.6 nM T75243 CPZ02V 132563118 IC50 = 114 nM T75243 C21KNJ 132563119 IC50 = 208 nM T75243 CT2PN8 132990561 IC50 = 16 nM T75243 C2AN7T 134611886 IC50 > 100000 nM T75243 CX0UR7 134694318 IC50 = 2920 nM T75243 C54FXD 134957362 IC50 > 10000 nM T75243 CT0GQ6 135197577 IC50 = 43 nM T75243 C87VKA 135197594 IC50 = 56 nM T75243 CQXS07 135197635 IC50 = 9.9 nM T75243 C7KXF1 135197643 IC50 = 7.9 nM T75243 CEK31P 135566415 IC50 > 20000 nM T75243 C24ZGX 135566644 IC50 > 10000 nM T75243 C2QDV5 135566741 IC50 > 10000 nM T75243 CU29YK 135750268 IC50 = 6000 nM T75243 CD6UJ5 135857414 IC50 = 1265 nM T75243 C41HNJ 135857415 IC50 = 170 nM T75243 CX4ZB3 135863110 IC50 = 18000 nM T75243 CRFO90 135870998 IC50 = 1020 nM T75243 CZ7Y0P 135871000 IC50 = 2880 nM T75243 C8K3HJ 135911704 IC50 = 23 nM T75243 C12UDA 135947972 IC50 = 3 nM T75243 CN42ZS 135947973 IC50 = 2100 nM T75243 CF8AO3 135947974 IC50 = 1130 nM T75243 CW08GJ 135947976 IC50 = 20 nM T75243 CJN7E2 135947978 IC50 = 1200 nM T75243 CFKH34 135947979 IC50 = 109 nM T75243 CXH63V 136041747 IC50 > 10000 nM T75243 C6B5TC 136041748 IC50 > 10000 nM T75243 CU6XG1 136041749 IC50 > 10000 nM T75243 C0U5DB 136041750 IC50 > 10000 nM T75243 C48KAQ 136041752 IC50 > 10000 nM T75243 C74PRL 136041753 IC50 > 10000 nM T75243 CCS2G6 136041761 IC50 > 10000 nM T75243 CEZP21 136041762 IC50 > 10000 nM T75243 CJ58TD 136041764 IC50 > 10000 nM T75243 CX67QW 136041765 IC50 > 10000 nM T75243 CK0H2Q 136041766 IC50 > 10000 nM T75243 CM65BS 136041773 IC50 > 10000 nM T75243 C6P7JB 136041775 IC50 > 10000 nM T75243 C5CJF7 136041776 IC50 > 10000 nM T75243 C3XIZ8 136041777 IC50 > 10000 nM T75243 C32LKO 136041785 IC50 > 10000 nM T75243 C90ARP 136041787 IC50 > 10000 nM T75243 CG19DI 136041799 IC50 > 10000 nM T75243 CS70RL 136042289 IC50 = 1270 nM T75243 CBHJ83 136042290 IC50 = 2440 nM T75243 C06KNL 136042291 IC50 = 630 nM T75243 CRA3T8 136042292 IC50 = 1050 nM T75243 CKT2U5 136042293 IC50 = 1930 nM T75243 CF3AV4 136042294 IC50 = 780 nM T75243 CZH70G 136042295 IC50 = 2380 nM T75243 CFN2U4 136042296 IC50 = 340 nM T75243 CK28EH 136042297 IC50 = 14100 nM T75243 CKE4R3 136042298 IC50 = 1670 nM T75243 CB0SV5 136042299 IC50 = 178 nM T75243 CQ0DF6 136042300 IC50 = 1040 nM T75243 C89CTO 136066004 IC50 = 32 nM T75243 CLA3C2 136068720 IC50 = 1200 nM T75243 C6ZH2F 136074294 IC50 = 2670 nM T75243 C1SME2 136074295 IC50 = 800 nM T75243 C95LGV 136074296 IC50 = 1940 nM T75243 CAK83X 136074297 IC50 = 6930 nM T75243 CTO47N 136079653 Ki = 2.9 nM T75243 CG1R7B 136087060 IC50 = 770 nM T75243 CC4UM3 136176116 IC50 > 10000 nM T75243 CJRK81 136176117 IC50 > 10000 nM T75243 C63IOS 136176118 IC50 > 10000 nM T75243 C3KW7H 136176119 IC50 > 10000 nM T75243 C69AKQ 136176120 IC50 > 10000 nM T75243 CF17KO 136176121 IC50 > 10000 nM T75243 CU3TE0 136176122 IC50 > 10000 nM T75243 C6C5KB 136176123 IC50 > 10000 nM T75243 C3X5KE 136176124 IC50 > 10000 nM T75243 CA8C5E 136176125 IC50 > 10000 nM T75243 C5OMG2 136176126 IC50 > 10000 nM T75243 CP2YM7 136176127 IC50 > 10000 nM T75243 C8XIJ0 136176128 IC50 > 10000 nM T75243 CUY8N4 136176129 IC50 > 10000 nM T75243 C3J4ME 136176130 IC50 > 10000 nM T75243 CR1NZ2 136176131 IC50 > 10000 nM T75243 C4WG2F 136176132 IC50 > 10000 nM T75243 CJ8EC5 136176139 IC50 > 10000 nM T75243 CHC5U8 136180788 IC50 = 550 nM T75243 C62SVA 136180789 IC50 = 560 nM T75243 C04XFY 136180790 IC50 = 52 nM T75243 CHLD54 136180791 IC50 = 550 nM T75243 CI6HG4 136249373 IC50 = 54 nM T75243 C0GZV9 136254283 IC50 > 10000 nM T75243 C3SJU4 136998793 IC50 = 2200 nM T75243 CH39TP 137453801 Ki = 137 nM T75243 C1EK8U 137453918 Ki = 37.9 nM T75243 CTZA58 137628643 IC50 = 7 nM T75243 C67EFJ 137628684 IC50 = 1.2 nM T75243 CZ5D6V 137631622 IC50 = 39.8 nM T75243 C1NWV2 137631657 IC50 = 222 nM T75243 CMI8E6 137632184 IC50 = 9.9 nM T75243 CN7WS0 137632234 IC50 = 75.8 nM T75243 CX39MO 137632259 IC50 = 31 nM T75243 C7Q2EY 137632337 IC50 = 70 nM T75243 CH8G2L 137632817 IC50 > 2000 nM T75243 CDEX29 137632839 IC50 > 2000 nM T75243 C38JDC 137633109 IC50 = 430 nM T75243 CZ7DR9 137633736 IC50 = 1190 nM T75243 CG73ZQ 137634050 IC50 > 2000 nM T75243 CTIA47 137634248 IC50 = 12 nM T75243 C5Z9FJ 137634261 IC50 = 425 nM T75243 CT40CM 137634322 IC50 > 2000 nM T75243 CCOG91 137634454 IC50 = 632 nM T75243 C6XMW2 137634650 IC50 = 410 nM T75243 CJN3B7 137634657 IC50 = 336 nM T75243 C34MHP 137634951 IC50 = 424 nM T75243 C8Q6WO 137635732 IC50 = 603 nM T75243 C7HBC4 137635822 IC50 = 4 nM T75243 CE4G3W 137635842 IC50 = 15.8 nM T75243 CHZ81K 137635885 IC50 = 104 nM T75243 C3KW5I 137636364 IC50 = 42 nM T75243 C5LHV9 137636943 IC50 = 29 nM T75243 C9UOW1 137637213 IC50 = 301 nM T75243 C5XKI7 137637306 IC50 > 2000 nM T75243 CU0O1W 137637367 IC50 = 422 nM T75243 CRP32A 137637486 IC50 > 2000 nM T75243 CSBY89 137637823 Ki = 660000 nM T75243 CMXV61 137637891 IC50 = 54.3 nM T75243 CO1V2E 137638253 IC50 > 2000 nM T75243 CS78JW 137639139 IC50 = 29000 nM T75243 C04NSI 137639729 IC50 = 26.2 nM T75243 CXZT29 137640462 Ki = 2539 nM T75243 CX1GO6 137641431 IC50 = 40.5 nM T75243 CJI94C 137641546 IC50 = 109 nM T75243 CG0FN1 137641601 IC50 = 167 nM T75243 C47VUG 137642023 IC50 = 54.9 nM T75243 CD2P5V 137642092 IC50 > 2000 nM T75243 CM1OD9 137642750 IC50 = 80 nM T75243 CP4DI5 137643070 IC50 = 330 nM T75243 C3QMK4 137643184 IC50 = 176 nM T75243 C4MVA7 137643536 IC50 > 2000 nM T75243 CUV1A4 137643705 IC50 = 55 nM T75243 C2ABR3 137644061 IC50 = 32 nM T75243 CL96JB 137644395 IC50 = 18.8 nM T75243 CP23NG 137644864 IC50 > 2000 nM T75243 C1O2NP 137645662 IC50 = 23 nM T75243 CI9D4L 137645884 IC50 = 290 nM T75243 CL4J3R 137646575 IC50 > 2000 nM T75243 CQ5T0F 137647241 IC50 = 24 nM T75243 CPMG65 137647250 IC50 = 10 nM T75243 CJ6KD5 137647435 IC50 = 865 nM T75243 C47HXI 137648104 IC50 = 1320 nM T75243 C7B6WC 137648193 IC50 = 4 nM T75243 CR9T0O 137648974 IC50 = 72.3 nM T75243 CK87YT 137649881 IC50 = 612 nM T75243 CECO31 137650069 IC50 = 463 nM T75243 CR6TM0 137650921 IC50 = 53 nM T75243 C7JQC2 137651055 Ki = 185 nM T75243 CI7R1A 137651064 IC50 = 32.9 nM T75243 CMV6K0 137651704 IC50 = 60 nM T75243 CF93QZ 137651837 IC50 = 3 nM T75243 C83KDE 137651894 IC50 = 172 nM T75243 C84TWB 137652545 IC50 = 73 nM T75243 CQMS19 137652991 IC50 > 2000 nM T75243 C5C7OQ 137653159 IC50 = 403 nM T75243 CN1P6C 137653212 IC50 = 201 nM T75243 C2LZE9 137653237 IC50 > 2000 nM T75243 CF4PA2 137654087 IC50 = 8.8 nM T75243 C2EVS5 137654553 IC50 > 2000 nM T75243 CPYL73 137654574 IC50 = 423 nM T75243 C7PF5R 137655359 IC50 = 82.9 nM T75243 C7ON1W 137655398 IC50 = 56 nM T75243 CD7X9E 137655716 IC50 = 3 nM T75243 CM26BD 137655969 IC50 = 14 nM T75243 C4VI2E 137656292 IC50 = 274 nM T75243 C0E8FC 137656416 IC50 = 40.6 nM T75243 CT9U7N 137656570 IC50 = 399 nM T75243 CCZ7P9 137656901 IC50 = 30.8 nM T75243 CA5ZU8 137657493 IC50 > 2000 nM T75243 CL8Z2V 137657573 IC50 = 36.6 nM T75243 CQE1B2 137657755 IC50 = 35 nM T75243 CX0NW5 137658179 IC50 = 3.57 nM T75243 CJ4QT6 137658610 IC50 = 335 nM T75243 C6MB1D 137658961 IC50 = 23.4 nM T75243 CWZ4P7 137659099 IC50 = 225 nM T75243 CT4CL9 137661232 IC50 = 3 nM T75243 CFJ5I9 137661497 IC50 = 427 nM T75243 CN73GX 137661561 IC50 > 2000 nM T75243 C81XWJ 137661590 Ki = 241 nM T75243 CZ25DA 137661970 IC50 = 68 nM T75243 CBS7L6 137662030 IC50 = 270 nM T75243 CA16BS 137662160 Ki = 110000 nM T75243 CA3C4O 138454792 IC50 = 2861 nM T75243 CKDZ26 138504497 IC50 = 5300 nM T75243 CDKR41 139030535 Ki = 8 nM T75243 C1NQ0F 139207772 Ki = 62 nM T75243 C3O5IA 139207773 Ki = 10 nM T75243 CKLH15 139207774 Ki = 4 nM T75243 C26NWP 139486659 Ki = 21.1 nM T75243 CV54CS 141471198 IC50 = 10 nM T75243 C25HYI 141471200 IC50 = 10 nM T75243 CZS03J 141509623 IC50 = 228 nM T75243 C8FZE6 142608579 Ki = 6 nM T75243 CR5GQ3 145949526 IC50 = 3450 nM T75243 C9E6AO 145950785 IC50 = 180 nM T75243 CDOU79 145953070 IC50 = 200 nM T75243 C7DO3I 145953589 IC50 > 10000 nM T75243 CG9F6T 145953725 IC50 = 90 nM T75243 CKQ63F 145955821 IC50 = 330 nM T75243 COC83T 145959468 IC50 = 260 nM T75243 C65YWX 145964882 IC50 > 10000 nM T75243 CHC3T0 145965031 IC50 > 10000 nM T75243 CP92ZF 145965329 IC50 > 10000 nM T75243 C9HXI4 145966620 IC50 > 10000 nM T75243 CQE9M5 145966810 IC50 > 10000 nM T75243 C1EH6C 145967078 IC50 > 10000 nM T75243 CWJ12M 145969155 IC50 > 10000 nM T75243 CGW5S1 145969844 IC50 > 10000 nM T75243 CB8R3A 145970271 IC50 > 10000 nM T75243 C40VIL 145972979 IC50 > 10000 nM T75243 CQBY19 145974023 IC50 > 10000 nM T75243 C4X7CT 145977420 IC50 > 10000 nM T75243 CLA57T 145978300 IC50 > 10000 nM T75243 CZ1T9X 145979969 Ki = 54.3 nM T75243 C03BJC 145980560 Ki = 3.4 nM T75243 CGA83C 145981271 IC50 = 34 nM T75243 CVR1X3 145981509 Ki = 60 nM T75243 CJ1G9L 145981832 Ki = 483 nM T75243 CH6X1R 145983184 Ki = 18.5 nM T75243 CD70WO 145986565 Ki = 435 nM T75243 CH7I9T 145987129 IC50 = 640 nM T75243 C5R6BS 145987142 IC50 = 52 nM T75243 C6D8QS 145987359 Ki = 474 nM T75243 C4BWJ3 145987648 Ki = 551 nM T75243 C9TYO4 145988008 Ki = 74.5 nM T75243 CACF81 145990005 IC50 = 720 nM T75243 C32MJQ 145990827 Ki = 79.9 nM T75243 CSYC93 145991982 Ki = 30 nM T75243 CA0J2B 145992083 Ki = 308 nM T75243 C36RTB 145993509 IC50 = 77.2 nM T75243 C4K0JW 145996540 IC50 = 21 nM T75243 CI85VS 146731761 IC50 = 9380 nM T75243 CLJ63X 147056594 IC50 > 1000 nM T75243 CT5HC9 147206876 IC50 > 1000 nM T75243 C7PI4F 147233226 IC50 = 253 nM T75243 C8TZB7 147371092 IC50 > 1000 nM T75243 CNA3L7 147416694 IC50 > 1000 nM T75243 CNAS83 147431947 IC50 = 48.6 nM T75243 CA21MO 147594782 IC50 > 1000 nM T75243 C05AJN 147697387 IC50 > 1000 nM T75243 CLH9U0 147709166 IC50 > 1000 nM T75243 CUQ8L3 147759183 IC50 = 17.9 nM T75243 CU72AS 147915791 IC50 > 1000 nM T75243 CA3TU9 147919900 IC50 = 267 nM T75243 C2J4TH 147979216 IC50 > 1000 nM T75243 C12CAJ 148039602 IC50 > 1000 nM T75243 CJ8NS7 148093822 IC50 > 1000 nM T75243 CSE50M 148120257 IC50 > 1000 nM T75243 CO0XB2 148191117 IC50 = 873 nM T75243 C5F3IQ 148239318 IC50 = 14.1 nM T75243 C92HBW 148300515 IC50 = 15.3 nM T75243 C74THK 148331443 IC50 > 1000 nM T75243 CZL64V 148493390 IC50 > 1000 nM T75243 CZ1N2T 148551789 IC50 > 1000 nM T75243 CND84O 148558668 IC50 > 1000 nM T75243 CWZ05D 148564044 IC50 = 13.85 nM T75243 CZA3D8 148695436 IC50 > 1000 nM T75243 CHER08 148928697 IC50 > 1000 nM T75243 CI8G9Y 149093021 IC50 = 34.9 nM T75243 CD2LF7 149098844 IC50 > 1000 nM T75243 CNY4Q3 149163842 IC50 = 19.4 nM T75243 COEI42 149296008 IC50 > 1000 nM T75243 CJ80FH 149323347 IC50 > 1000 nM T75243 CN87RZ 149370890 IC50 > 10000 nM T75243 C82BFC 149396423 IC50 > 1000 nM T75243 COMP43 149503998 IC50 > 1000 nM T75243 CK4FJ1 149556361 IC50 = 8120 nM T75243 C2ABX3 152981558 IC50 = 19.8 nM T75243 C7ZU5T 153109924 IC50 = 13.8 nM T75243 C6RFV3 153244706 IC50 > 1000 nM T75243 CU42HJ 153248266 IC50 = 12.6 nM T75243 CJ0EN5 153262665 IC50 > 1000 nM T75243 C8UQL4 153940691 IC50 > 10000 nM T75243 CMZ68Q 153940692 IC50 > 10000 nM T75243 CY2WZ6 155233745 IC50 = 256.8 nM T75243 CDXM69 155249380 IC50 = 7766 nM T75243 CH6V0O 155249545 IC50 = 29.24 nM T75243 C1OVC9 155511557 Ki = 2.5 nM T75243 CG49LC 155512502 IC50 = 3.1 nM T75243 CG9I4X 155512515 IC50 = 7440 nM T75243 CR1Z8A 155512529 IC50 = 5300 nM T75243 C2MD1Q 155513187 IC50 > 10000 nM T75243 CF6CG8 155513897 IC50 > 1000 nM T75243 C17NTI 155514706 Ki = 2200 nM T75243 CEFS61 155515135 IC50 > 10000 nM T75243 CX72DF 155515279 IC50 = 5011.87 nM T75243 CBK3C9 155515384 Ki = 20 nM T75243 CI50FQ 155516321 IC50 > 1000 nM T75243 C8FWK7 155517588 IC50 = 501.19 nM T75243 C5D6YX 155521099 IC50 > 10000 nM T75243 CC1P7U 155521604 IC50 > 1000 nM T75243 CABC57 155522182 Ki = 1700 nM T75243 C5AHS1 155523025 IC50 = 4.3 nM T75243 CZ3FC8 155523374 Ki = 43.1 nM T75243 CZG27I 155523570 IC50 = 676 nM T75243 CG61OL 155524143 IC50 > 1000 nM T75243 CJMD34 155525139 Ki = 190 nM T75243 C9E2PJ 155525385 IC50 = 290.5 nM T75243 C3I9UX 155526450 Ki = 27 nM T75243 CPJ3R6 155526809 Ki = 9.1 nM T75243 C9PF1D 155527778 IC50 = 635 nM T75243 CF2P3Q 155527936 Ki = 1892 nM T75243 CJ3LP5 155528779 Ki = 56 nM T75243 C9OVL5 155528904 Ki = 50 nM T75243 CNA30V 155529246 IC50 > 1000 nM T75243 C9L6OC 155529247 IC50 = 6262 nM T75243 CPH72K 155531472 IC50 > 1000 nM T75243 CA7T0Y 155533911 IC50 > 10000 nM T75243 C68NQP 155536585 Ki = 96 nM T75243 C1Y9MS 155537503 Ki = 2300 nM T75243 CHR8M1 155538990 IC50 = 9120 nM T75243 CE8TV9 155541005 Ki = 40 nM T75243 CN5U9M 155541206 Ki = 34 nM T75243 CYB90C 155542790 Ki = 4000 nM T75243 C8OC2P 155542800 IC50 = 660 nM T75243 CV5L6B 155543139 Ki = 370 nM T75243 CBN29V 155544583 IC50 = 846 nM T75243 C5IVX6 155544961 Ki = 265 nM T75243 CV9OI5 155545359 IC50 = 3.6 nM T75243 CE02BC 155545624 IC50 = 1584.89 nM T75243 CJ1E0T 155547067 Ki = 59.2 nM T75243 CKR36G 155547524 Ki = 39.6 nM T75243 C6JCV4 155548973 Ki = 13 nM T75243 CJWV35 155549094 Ki = 33 nM T75243 C4PEJ5 155549895 IC50 > 10000 nM T75243 CGNF42 155549917 Ki = 76.8 nM T75243 CQ5OD0 155550395 IC50 = 181 nM T75243 CE5DG7 155550972 Ki = 104 nM T75243 CVO9N5 155551369 Ki = 208 nM T75243 CF8D9H 155552080 Ki = 47.8 nM T75243 CJ75BO 155552100 IC50 = 6550 nM T75243 C8L4MZ 155554924 Ki = 85 nM T75243 CCY47Q 155554935 IC50 > 1000 nM T75243 CFW90N 155555562 IC50 = 40 nM T75243 C3BK7O 155556309 Ki = 171 nM T75243 CO4GE3 155557022 Ki = 31 nM T75243 C0FE4G 155557988 IC50 > 10000 nM T75243 C6BAV3 155558720 Ki = 24 nM T75243 CZCO50 155559160 Ki = 300 nM T75243 C7TP0F 155559332 Ki = 60 nM T75243 CVG49I 155560688 IC50 > 10000 nM T75243 C4GXV3 155562151 Ki = 28 nM T75243 C6RV0H 155563416 Ki = 11 nM T75243 CTEB79 155563891 Ki = 31 nM T75243 CC04GI 155564488 IC50 = 31.62 nM T75243 C5SH4P 155565730 Ki = 121 nM T75243 CPA75N 155566172 IC50 = 3.4 nM T75243 C3XMB6 155567232 Ki = 21 nM T75243 C1S8ZB 155568922 IC50 = 3450 nM T75243 CTG81X 155569017 Ki = 177 nM T75243 CUH38L 155569363 IC50 = 8370 nM T75243 CVR2J1 155569607 Ki = 13 nM T75243 D00GQM 25069592 IC50 = 4500 nM T75243 D00JIV 51033720 Ki = 1440 nM T75243 D02TCF 44576240 IC50 = 5 nM T75243 D02TSN 46244454 IC50 = 38 nM T75243 D03EHM 24905142 IC50 = 10 nM T75243 D03QQH 16760391 IC50 > 100000 nM T75243 D05BPX 9901372 IC50 = 49 nM T75243 D05USL 5278396 IC50 = 5580 nM T75243 D06HVH 54613583 IC50 > 9100 nM T75243 D07JKB 135955185 IC50 = 2500 nM T75243 D07PMP 44187953 IC50 = 1.7 nM T75243 D09FBN 135955186 IC50 = 450 nM T75243 D0AH8Q 25074311 IC50 = 2800 nM T75243 D0F1SI 25074312 IC50 = 3900 nM T75243 D0H0HR 49836027 IC50 = 4.32 nM T75243 D0H2CM 135565635 IC50 = 8 nM T75243 D0R0TW 11964036 IC50 = 10000 nM T75243 D0T0BY 10039361 IC50 = 5300 nM T75243 D0TC5H 16049458 IC50 = 1650 nM T75243 D0U8GR 44576241 IC50 = 10 nM T75243 D0W1ST 9860529 IC50 = 6400 nM T75243 D0W8XH 9884685 IC50 = 8.8 nM T75243 D0X7TB 10017389 IC50 = 4800 nM T75243 D0Y1DR 46225260 IC50 = 150 nM T75243 D0Y3OO 11327430 IC50 = 1700 nM T35194 CSAL71 1139373 IC50 = 19000 nM T35194 C60KGD 1139434 IC50 = 35000 nM T35194 CR2Q7B 1276013 IC50 = 25000 nM T35194 CW82ZQ 1336260 IC50 = 11000 nM T35194 CX3YR6 1349305 IC50 = 16000 nM T35194 CY4O7M 1718303 IC50 = 2700 nM T35194 CEP6M9 2279002 IC50 = 17000 nM T35194 CTD14H 2281496 IC50 = 6600 nM T35194 C0PCZ3 5932584 IC50 = 520 nM T35194 CU65JT 5998084 IC50 = 780 nM T35194 C14LAC 6161281 IC50 = 460 nM T35194 CR6O8V 6166563 IC50 = 2800 nM T35194 CYI5R1 6274486 IC50 = 470 nM T35194 C4JTB5 6419844 IC50 = 11500 nM T35194 C5GRL3 17103728 IC50 = 27000 nM T35194 CKP32L 21211508 IC50 = 17000 nM T35194 C4INO9 22776482 IC50 = 21000 nM T35194 C2V7NL 135797380 IC50 > 100000 nM T35194 C27EYJ 135797381 IC50 > 100000 nM T35194 CZOL36 135797386 IC50 > 100000 nM T35194 CBX75S 135797387 IC50 > 100000 nM T35194 C2L6UZ 135797388 IC50 > 100000 nM T35194 C0S1VO 135797389 IC50 > 100000 nM T35194 CS40TI 135797392 IC50 > 100000 nM T35194 C0RJW6 135797397 IC50 > 100000 nM T35194 C5UL0V 135955126 IC50 > 100000 nM T35194 C85VGD 136069445 IC50 > 100000 nM T35194 CQ7L2H 136254273 IC50 > 100000 nM T35194 C5C1XF 136254274 IC50 > 100000 nM T35194 CL4A5E 136254275 IC50 > 100000 nM T35194 CH7N3Z 136254276 IC50 > 100000 nM T35194 CL4ZM7 136254277 IC50 > 100000 nM T35194 CAHC90 136254278 IC50 > 100000 nM T35194 CQ84LN 136254279 IC50 > 100000 nM T35194 CBEU97 136254280 IC50 > 100000 nM T35194 C3LK1C 136254281 IC50 > 100000 nM T35194 C5RF9N 155524598 IC50 = 16000 nM T35194 CD19LB 155526448 IC50 = 4800 nM T35194 C5GLU2 155529287 IC50 = 8300 nM T35194 CA93NV 155541948 IC50 = 7900 nM T35194 C6JV0T 155551451 IC50 = 8700 nM T63068 D0D8VE 3562 IC50 = 2900000 nM T63068 CFU83O 9898808 IC50 = 1200000 nM T63068 CWP0A7 9990042 IC50 = 400000 nM T63068 C5RM3V 10036388 IC50 = 800000 nM T63068 CSJ8W7 10944023 IC50 = 300000 nM T63068 C7RB3E 11041260 IC50 = 2200000 nM T63068 C2PW6B 11075469 IC50 = 700000 nM T63068 C4Z7CN 25100119 Ki = 400 nM T63068 CHYW16 25144061 Ki = 360 nM T63068 CQ2RZ7 25144887 Ki < 30 nM T63068 C6K8UH 44356682 IC50 = 23000 nM T63068 C8RK3T 54678499 Ki = 3300 nM T63068 C5M4OJ 68940388 Ki = 1450 nM T63068 CF4G5B 118734953 Ki > 100000 nM T20401 D00STL 644241 Ki = 4.1 nM T20401 D00ZOF 23666456 Ki = 3220000 nM T20401 D01MUR 68844 Ki = 0.1259 nM T20401 D01WJL 4649 IC50 = 750000 nM T20401 D02FLB 516892 Ki = 85000000 nM T20401 D02PJA 24841 Ki = 26000000 nM T20401 D02URS 4875 Ki = 26000000 nM T20401 D02ZTJ 5339 IC50 = 4490 nM T20401 D03QGM 5355 Ki = 40 nM T20401 D03RTS 2662 Ki = 21 nM T20401 D03UOT 785 Ki = 90 nM T20401 D04AIT 5280445 Ki = 3691.6 nM T20401 D04YZL 5234 Ki = 200000000 nM T20401 D05OFX 219078 Ki = 331 nM T20401 D05UYW 5284549 IC50 = 0.18 nM T20401 D05VGL 11499245 Ki = 462 nM T20401 D07CWD 3657 Ki = 28000 nM T20401 D07HBX 338 Ki = 7100 nM T20401 D07INV 3295 Ki = 0.49 nM T20401 D07MGA 72281 Ki > 10000 nM T20401 D07VDZ 5284627 Ki = 5 nM T20401 D08LFZ 3059 IC50 = 2700 nM T20401 D09NIA 2732 Ki = 138 nM T20401 D09VAZ 5565 Ki = 64000 nM T20401 D0A3HB 4943 Ki = 19500 nM T20401 D0AZ3C 5291 Ki = 30.2 nM T20401 D0AZ8C 5213 Ki = 2510 nM T20401 D0C2II 4100 Ki = 9 nM T20401 D0C8EU 5394 Ki > 50000 nM T20401 D0C8FX 3005837 Ki > 200000 nM T20401 D0E1SW 1986 Ki = 0.012 nM T20401 D0E9JM 4873 Ki > 200000000 nM T20401 D0GY5Z 2244 IC50 = 1160000 nM T20401 D0H8FH 3702 Ki = 2520 nM T20401 D0J4GO 3038 Ki = 8 nM T20401 D0J7RK 36811 Ki = 480 nM T20401 D0K0OZ 5702160 Ki = 57.9 nM T20401 D0K1QD 3998 Ki = 170 nM T20401 D0K8KX 5280343 Ki = 2540 nM T20401 D0L4JT 5333 Ki = 240 nM T20401 D0L6DA 119607 IC50 = 43 nM T20401 D0L7FM 4911 Ki = 431 nM T20401 D0MA7C 23668193 Ki = 63000000 nM T20401 D0MD2L 129228 Ki > 10000 nM T20401 D0OT0O 44561 Ki = 14200000 nM T20401 D0PQ3G 3440 Ki = 65 nM T20401 D0R0FO 9823820 Ki > 10000 nM T20401 D0R9BG 1990 IC50 = 47000 nM T20401 D0SH3I 387447 Ki = 1160 nM T20401 D0TG1H 3033 IC50 > 100000 nM T20401 D0U4UQ 3639 Ki = 290 nM T20401 D0U5QK 1983 Ki = 6200 nM T20401 D0V8QT 2708 Ki > 50000 nM T20401 D0VM2L 68740 IC50 = 62 nM T20401 D0W5HK 216239 Ki > 10000 nM T20401 D0Y2IZ 5560 Ki = 91 nM T20401 D0Z3EI 6038 Ki > 10000 nM T20401 D0Z4UY 517045 Ki = 130000 nM T20401 D02ECG 23662274 Ki = 2110000 nM T20401 D02JUW 460 Ki = 2940 nM T20401 D04IIU 216468 IC50 = 15 nM T20401 D04PBH 5280804 Ki = 410 nM T20401 D05NJI 5287541 IC50 = 17 nM T20401 D05ZXZ 491941 Ki = 12.8 nM T20401 D06DMQ 59472121 Ki > 50000 nM T20401 D06PII 5356 Ki = 9 nM T20401 D07ZNI 9804302 Ki = 270 nM T20401 D08BXT 1102 Ki = 1110 nM T20401 D09XQU 135413511 Ki > 50000 nM T20401 D0C2KF 11616111 IC50 = 5000 nM T20401 D0I7IB 5222465 Ki = 1032000 nM T20401 D0I7MT 5281807 Ki > 10000 nM T20401 D0L6HN 996 Ki = 5500 nM T20401 D0SC6I 517055 Ki = 30000 nM T20401 D0TO2R 30751 Ki > 10000 nM T20401 D0U3EP 445154 Ki = 2770 nM T20401 D0V0UK 82267 Ki = 1.13 nM T20401 D0W1SL 31404 Ki = 630 nM T20401 D03SLR 445858 Ki = 2400 nM T20401 D08RPE 71607911 IC50 > 10000 nM T20401 D0F8XZ 19890 Ki > 100000 nM T20401 D0NH9P 135 Ki = 870 nM T20401 D0X2AU 23427 Ki > 100000 nM T20401 D07XPE 8249 Ki > 50000 nM T20401 D0LD9S 1103 Ki = 84000 nM T20401 CI0WH9 72 Ki = 470 nM T20401 CJ28SX 127 Ki = 10300 nM T20401 CUT2V4 260 Ki = 63000000 nM T20401 COV5W3 402 Ki = 2800 nM T20401 CSZ43B 540 Ki = 30000 nM T20401 C97QXH 767 Ki = 73000000 nM T20401 C39CTO 768 Ki = 20000 nM T20401 C1QDT0 781 Ki = 1600000 nM T20401 CAD4R0 798 Ki = 32500 nM T20401 CW0R2L 944 Ki = 35000000 nM T20401 C2LNM9 1016 Ki = 1080000 nM T20401 C6QX8I 1089 Ki = 112000000 nM T20401 CQV86E 1100 Ki = 89000000 nM T20401 C8W7BZ 1118 Ki = 89000000 nM T20401 CU12QE 1203 Ki = 1840 nM T20401 C6O0MZ 1491 Ki = 4900 nM T20401 C49BCY 1570 Ki = 510000 nM T20401 CO4X7B 2456 Ki = 395 nM T20401 C5L7VX 2871 Ki > 200000 nM T20401 CZP5J2 3415 Ki = 14200000 nM T20401 CQ0D8J 3469 Ki = 4100 nM T20401 CJ2F6P 5056 Ki = 1750 nM T20401 CTDR62 5235 Ki > 200000000 nM T20401 CKQC48 5238 Ki = 26000000 nM T20401 CRAO91 5324 IC50 > 100000 nM T20401 CDJ4K6 5987 Ki = 0.39 nM T20401 CGTE42 6101 Ki = 460000 nM T20401 CU9EM3 6125 Ki = 990000 nM T20401 C4V7LO 6738 IC50 = 4700000 nM T20401 CUP2F4 7043 Ki = 500 nM T20401 C1CVT7 7121 Ki = 6180 nM T20401 CHG8L5 7322 IC50 = 290000 nM T20401 C6NC4O 7414 Ki = 51000 nM T20401 CJKY76 7420 Ki = 600 nM T20401 C23KMD 7921 Ki > 100000 nM T20401 C6QYD8 8434 Ki = 4800 nM T20401 CD6O9A 8499 Ki = 3530 nM T20401 C46OQB 8697 Ki = 93000 nM T20401 CXF7C6 8736 Ki = 1870000 nM T20401 CR3IF4 8865 Ki = 1620000 nM T20401 C8VKM7 8929 Ki = 20000 nM T20401 C40HCL 8987 Ki = 3100000 nM T20401 CHP7I1 9016 Ki = 3350 nM T20401 CLYZ50 9338 Ki = 5200 nM T20401 CNM7L3 10199 Ki > 10000 nM T20401 CBIR94 10313 Ki = 179000 nM T20401 COU60V 10340 Ki = 73000000 nM T20401 CC30SK 10341 Ki > 100000 nM T20401 CM20CY 10393 Ki = 8700 nM T20401 C4NQE7 10787 Ki > 100000 nM T20401 CACI42 10953 Ki > 100000 nM T20401 C7H1FT 11335 Ki = 113500 nM T20401 CUG8B9 11418 Ki = 340 nM T20401 CCPT31 11419 Ki = 420 nM T20401 CV5PC3 11568 Ki = 4700 nM T20401 CL80QG 11820 Ki > 10000 nM T20401 C14BYX 12662 Ki > 100000 nM T20401 C57OTC 13818 Ki = 98 nM T20401 CKA21F 14768 Ki = 2680000 nM T20401 CUA0L6 14917 Ki > 300000000 nM T20401 CNI85U 15109 Ki = 1020 nM T20401 CS8X0P 16124 Ki = 1250000 nM T20401 CQ4C5U 16523 Ki = 760 nM T20401 CS39YR 19654 Ki = 850000 nM T20401 CNGB21 20098 Ki = 660 nM T20401 C7OJ9Q 20125 Ki = 3450 nM T20401 C3LA1Z 20161 Ki = 4400 nM T20401 CMK0O4 20825 Ki > 10000 nM T20401 CF14KR 24247 Ki = 1260000 nM T20401 CHW5M0 24268 Ki = 35000000 nM T20401 C4IZB8 24345 Ki = 48900000 nM T20401 CGR6D5 24413 Ki = 84000 nM T20401 C9M8EJ 24434 Ki = 35000000 nM T20401 CAN29U 24436 Ki > 200000000 nM T20401 C8S9AF 24445 Ki = 12000000 nM T20401 C3NG2U 24529 Ki = 63000000 nM T20401 CFM9L6 24530 Ki = 1500000 nM T20401 CBT68I 24603 Ki = 460000 nM T20401 C3F1OY 25502 Ki = 830000 nM T20401 CF2XP3 26255 Ki > 200000000 nM T20401 CG04AY 26518 Ki = 1720 nM T20401 CDK20Z 27290 Ki = 2600 nM T20401 CWIZ67 28015 Ki = 40000 nM T20401 C69RDT 32204 Ki = 7510 nM T20401 C7YZM4 33557 Ki = 1500000 nM T20401 C4OU6D 35703 Ki = 161000 nM T20401 CDIJ43 36573 Ki > 20000 nM T20401 C89DPG 39981 Ki = 7800 nM T20401 CY2GU3 60582 Ki = 18.2 nM T20401 CR5W8Y 60692 Ki = 0.7 nM T20401 CT26XL 60693 IC50 = 0.54 nM T20401 C1N6SE 61127 Ki = 29820 nM T20401 CF26VS 61441 Ki = 510000 nM T20401 C6R1AJ 61609 Ki = 920000 nM T20401 CLMR98 61857 Ki = 6230000 nM T20401 CJ03HR 62481 Ki = 1600000 nM T20401 CV28FU 62805 Ki > 10000 nM T20401 C5MJH8 64789 Ki > 50000 nM T20401 CKQA52 64999 Ki = 140 nM T20401 CN94KU 65008 Ki = 50700 nM T20401 C6DG9Q 65185 Ki = 75800000 nM T20401 C1NQ8E 65188 Ki > 100000 nM T20401 CT6YO0 66548 Ki > 100000 nM T20401 CCE63L 66634 IC50 = 808.81 nM T20401 CMXS19 66814 Ki = 3333.8 nM T20401 CJ1Z2R 67125 Ki = 4190 nM T20401 C0ZK7U 67284 Ki = 1430 nM T20401 C8H4AT 67313 Ki = 25000 nM T20401 CWXE69 67756 Ki = 378 nM T20401 C26PTJ 67760 Ki = 642 nM T20401 CJWD84 68154 Ki > 100000 nM T20401 CA3R7P 68351 Ki = 6 nM T20401 CB89AL 68982 Ki = 8800 nM T20401 CYEU83 69033 Ki = 26 nM T20401 CC0R8X 69696 Ki = 81 nM T20401 CVI38F 69809 Ki = 66300 nM T20401 CND3B8 70122 Ki = 166400 nM T20401 CX4HM3 70653 IC50 = 3623 nM T20401 CI80QC 71485 Ki = 300 nM T20401 C8U0VH 72597 Ki = 0.92 nM T20401 CJR96B 72879 Ki = 390000 nM T20401 CU79WI 74093 Ki = 2 nM T20401 CTMF08 75076 Ki = 690 nM T20401 C0I4UT 75077 Ki = 770 nM T20401 C7L1RO 75522 Ki = 638 nM T20401 CE5RZ1 76509 Ki = 11200 nM T20401 C8DHG4 76792 Ki = 5750 nM T20401 CXG7Y0 76959 Ki = 2180 nM T20401 CVSE97 77456 Ki = 8560 nM T20401 C9V0ME 77547 Ki = 610 nM T20401 C6TS8J 77548 Ki = 690 nM T20401 CRXH06 77553 Ki > 10000 nM T20401 CZAX86 77578 Ki = 57500 nM T20401 C0PY5N 77754 Ki = 4.7 nM T20401 CX79KD 78297 Ki = 39.5 nM T20401 CX47BZ 78479 Ki = 75000 nM T20401 C1TJF6 79001 Ki = 2 nM T20401 CCK8E1 79611 Ki = 10.1 nM T20401 C9QAS6 86986 Ki = 11200 nM T20401 C5BFK4 87432 Ki = 2820 nM T20401 CYIP60 89607 Ki = 50 nM T20401 CM72DQ 90631 Ki = 240 nM T20401 CB5R7Y 92229 Ki > 100000 nM T20401 CB81UG 93577 Ki = 77000 nM T20401 CJ01AO 94706 Ki = 7 nM T20401 C2GI9X 95801 IC50 > 50000 nM T20401 C40RWH 95840 Ki = 86 nM T20401 C21JNS 95841 Ki > 10000 nM T20401 C5Z1QA 96028 IC50 > 200000 nM T20401 C1GQE3 97576 Ki = 3410 nM T20401 CEC01M 97598 Ki = 2360 nM T20401 CSGF32 99327 Ki = 103900 nM T20401 CA9YN2 99477 Ki > 10000 nM T20401 CV76MT 100187 Ki > 50000 nM T20401 CGM6A9 101263 Ki > 1000 nM T20401 C6K3MG 101424 Ki > 100000 nM T20401 C9Q4GE 102491 Ki = 2050 nM T20401 CI8DH1 103993 Ki > 10000 nM T20401 CD48YU 108326 Ki = 17 nM T20401 C27CDU 118534 Ki = 8600 nM T20401 CP4O2C 121255 Ki = 18 nM T20401 CK3C4Q 121595 IC50 = 5 nM T20401 CDP5M6 125623 Ki = 65.2 nM T20401 C4MO7F 126061 IC50 = 4 nM T20401 CN19UT 129695 Ki = 1130 nM T20401 CUX39B 132037 Ki = 1130 nM T20401 CCK5Y6 133125 Ki = 8.1 nM T20401 CVB67D 134560 Ki = 2 nM T20401 CYH75F 135214 IC50 = 40 nM T20401 CD2HC7 138614 Ki = 380 nM T20401 C2P0RH 139584 Ki = 750000 nM T20401 CUBQ92 145746 Ki = 5500 nM T20401 C5GMZ4 146921 IC50 = 8.8 nM T20401 C9ZEP5 151399 Ki > 10000 nM T20401 C47BCV 154989 Ki = 417 nM T20401 CJ0FR9 155148 Ki = 49300 nM T20401 C50XVJ 159772 Ki = 1150 nM T20401 C1SAJ0 162152 Ki = 760000 nM T20401 CW2Y7L 162287 Ki > 10000 nM T20401 CVH81Y 163571 Ki = 133 nM T20401 C4U5KL 164000 IC50 = 720000 nM T20401 C8AO0Z 165323 Ki = 12 nM T20401 C6M0TK 167985 Ki = 760000 nM T20401 CU3WG6 179620 Ki > 100000 nM T20401 CE1VJ6 191826 Ki > 100000 nM T20401 CO96LR 192271 Ki = 7 nM T20401 C60KJD 192792 Ki = 131 nM T20401 CB34GS 195580 Ki = 1.58 nM T20401 C1N3AY 199210 Ki = 3690 nM T20401 C2GHM7 202375 IC50 = 6672 nM T20401 CSMP84 219987 Ki = 135000 nM T20401 C9K3VU 220023 IC50 > 50000 nM T20401 C90VSK 221131 Ki = 450 nM T20401 CEZU63 221227 Ki = 3420 nM T20401 C5CQ1I 222870 Ki = 29.51 nM T20401 C7DS2I 228958 Ki = 41.5 nM T20401 C2ED9N 236541 Ki > 10000 nM T20401 C14USE 239728 Ki > 50000 nM T20401 CW1E5G 239730 Ki = 1260 nM T20401 CP7Q8T 240910 Ki = 37 nM T20401 CRP27E 245904 Ki = 63 nM T20401 C6D1LY 246499 Ki = 166 nM T20401 C0B3OQ 253877 Ki = 63000000 nM T20401 C6DQU8 253881 Ki = 63000000 nM T20401 CLV79E 260228 Ki = 3600 nM T20401 CU45WA 260244 Ki > 100000 nM T20401 CI83OK 273360 Ki = 18310 nM T20401 C0UL5Y 276741 Ki = 148 nM T20401 CX3DK6 283995 Ki = 29 nM T20401 C1QOB5 284045 Ki = 59107 nM T20401 C3QV5H 287064 Ki = 580 nM T20401 C26HNY 289493 Ki = 63400 nM T20401 C51UMX 294719 Ki = 54 nM T20401 C83MLQ 295450 Ki = 1800 nM T20401 COE9A7 306924 Ki = 240 nM T20401 CAUO79 306968 Ki = 33 nM T20401 CM2N3X 307505 Ki = 10 nM T20401 C3W0AQ 307522 Ki = 4070 nM T20401 C3WZI1 308397 Ki = 258 nM T20401 C6AKQ8 308411 Ki = 328 nM T20401 CL4GF1 308432 Ki = 290 nM T20401 C96DKW 310360 Ki = 96 nM T20401 CY13EN 311156 Ki = 276 nM T20401 C12PJC 313721 IC50 = 7321 nM T20401 CQ67ZL 315810 Ki = 133 nM T20401 COI7H8 317746 Ki = 15.6 nM T20401 CG3J6Q 323350 Ki = 2.3 nM T20401 CTX0Z3 327169 Ki > 100000 nM T20401 C8K5LE 338294 Ki > 10000 nM T20401 CXZ14S 341082 Ki > 50000 nM T20401 CP7X9H 342056 Ki > 10000 nM T20401 CMS5W4 343662 Ki > 10000 nM T20401 C5V2ZH 345312 Ki = 10 nM T20401 CH1C9B 351361 Ki > 1000 nM T20401 COFX01 352863 Ki = 21 nM T20401 CM9V8O 388547 Ki > 10000 nM T20401 CT3ZU4 388776 Ki = 11300 nM T20401 CH21KA 389641 Ki = 107000 nM T20401 C6CQO3 389642 Ki = 110000 nM T20401 CH0F9P 390929 Ki = 158 nM T20401 CNPZ40 394897 Ki = 10 nM T20401 C4WC2P 394900 Ki = 10 nM T20401 CY39DK 394901 Ki = 9 nM T20401 CGUJ45 394902 Ki = 6 nM T20401 C2G6DI 394904 Ki = 4 nM T20401 C9NF6V 395814 Ki = 100 nM T20401 CHU17A 395815 Ki = 3 nM T20401 C5TON3 395826 Ki = 4 nM T20401 CL5WQ3 396510 Ki = 12 nM T20401 C10GOE 397555 IC50 = 7 nM T20401 C7HME8 439246 Ki > 10000 nM T20401 CA8C5N 439514 Ki > 100000 nM T20401 C3W8LP 445393 Ki = 12 nM T20401 CC54LQ 450256 IC50 > 10000 nM T20401 C5IPL1 471796 Ki = 4860 nM T20401 C5HM8E 474578 Ki = 127 nM T20401 CU53VO 482060 Ki = 660 nM T20401 CL0M9Y 482317 Ki = 3920 nM T20401 CHF2Y9 493949 Ki = 361 nM T20401 C9YHN5 499219 Ki = 2300000 nM T20401 C02DMG 504302 Ki = 4.9 nM T20401 CU7XE2 504303 Ki = 180 nM T20401 CNLT49 504304 Ki = 248 nM T20401 COGF52 516871 Ki = 200000 nM T20401 CC2V0U 517096 Ki = 30000 nM T20401 CD8S2T 517441 Ki = 8130 nM T20401 C49CNT 519869 Ki = 700 nM T20401 C49LCW 519974 Ki > 100000 nM T20401 CU8MR5 520660 Ki > 100000 nM T20401 CQK9J0 522606 Ki > 100000000 nM T20401 C5OA7L 522689 Ki > 300000000 nM T20401 CJ7FR6 533728 Ki = 3100 nM T20401 C24ASH 539731 Ki = 55.5 nM T20401 C7EBA4 540544 Ki > 10000 nM T20401 CFU6X9 560256 Ki = 6910 nM T20401 C3H5SW 562880 Ki = 56400 nM T20401 CPV28T 567846 Ki = 82 nM T20401 CU83WT 587961 Ki = 38000 nM T20401 CGHE12 607195 Ki = 2210 nM T20401 CIK9S3 607305 Ki > 10000 nM T20401 CP3SF2 609637 Ki = 59 nM T20401 C5EA3O 638001 Ki > 100000 nM T20401 CNR94Z 640087 IC50 = 23140 nM T20401 C1DX6J 640625 Ki > 100000 nM T20401 CUMO27 643477 Ki > 100000 nM T20401 C58QOW 643497 Ki = 40 nM T20401 CH05FZ 648662 Ki > 10000 nM T20401 C6PTC3 658040 Ki > 50000 nM T20401 CRZB53 669716 Ki = 127 nM T20401 CU9ZY6 670087 Ki = 104 nM T20401 CYGK68 676946 Ki = 710 nM T20401 CMO61A 694792 Ki = 52 nM T20401 CF9V6Q 699414 IC50 = 760000 nM T20401 C4YWI2 702292 Ki = 190 nM T20401 CYZ9O5 703304 Ki > 10000 nM T20401 C9JH0M 706033 Ki = 42 nM T20401 C7ZE6K 706849 Ki > 50000 nM T20401 CK7DO5 708535 Ki = 28 nM T20401 CK9HY0 716763 Ki > 1000 nM T20401 C8J4SO 724642 Ki = 40 nM T20401 C61NGE 724799 Ki = 5 nM T20401 CNTI96 728666 Ki = 97400 nM T20401 C8J7CO 730546 Ki = 14.2 nM T20401 C8G7EC 730672 Ki = 781 nM T20401 COQ14K 738631 Ki = 7 nM T20401 CNJZ35 738819 Ki > 50000 nM T20401 CV6Y7U 740560 IC50 > 50000 nM T20401 CZM6W0 742873 Ki = 4.8 nM T20401 C3SAH9 743904 Ki = 9 nM T20401 CLG6H5 746816 Ki > 1000 nM T20401 CRIJ01 747569 Ki = 53 nM T20401 C61BMV 751041 Ki = 19320 nM T20401 CW90GV 767467 Ki > 1000 nM T20401 CV79DU 776418 Ki > 50000 nM T20401 CQJ06V 780268 IC50 = 60.93 nM T20401 CO1KN3 788171 Ki = 5.5 nM T20401 CA2B8X 792066 Ki = 404 nM T20401 CM0VX3 809685 Ki = 3.5 nM T20401 CT0WB5 810867 Ki > 100000 nM T20401 C6LN8S 816982 Ki > 500000 nM T20401 C5BGW9 818267 Ki > 50000 nM T20401 CJP5D4 818647 IC50 = 5100 nM T20401 CVJZ57 818753 Ki > 50000 nM T20401 CF93TC 821388 Ki = 520 nM T20401 C5VJZ0 822776 Ki = 0.79 nM T20401 CTD64N 834412 Ki = 1.8 nM T20401 CHE97G 834460 IC50 = 12.54 nM T20401 CO31FL 853546 Ki = 123.2 nM T20401 C8SN5L 889524 Ki = 33.8 nM T20401 CQ45SF 892618 Ki = 42 nM T20401 CEN67I 897592 Ki = 2810 nM T20401 C51FVL 906840 Ki > 10000 nM T20401 CL2G3R 917163 Ki = 13 nM T20401 CKV7B6 917551 Ki > 10000 nM T20401 C4I3PJ 922062 Ki = 7.4 nM T20401 CRGQ70 927433 Ki > 200000 nM T20401 CO7XW0 928228 Ki > 10000 nM T20401 C6XQO2 940540 Ki > 50000 nM T20401 C4L9QD 943114 Ki > 10000 nM T20401 COH62A 943115 Ki > 10000 nM T20401 C7FI1J 970570 Ki = 45 nM T20401 CX3U0S 975396 Ki > 50000 nM T20401 CZ3WK7 983751 Ki > 1000 nM T20401 CN71CV 989611 Ki > 10000 nM T20401 C4TE0N 990581 Ki = 123 nM T20401 C5CED0 1014382 IC50 = 11.82 nM T20401 CXQ3M7 1016209 IC50 = 41.97 nM T20401 C6MU1W 1069008 Ki = 5 nM T20401 CJ2S0M 1070919 Ki = 14.3 nM T20401 CYS9A2 1070922 Ki = 6.9 nM T20401 CM2C5N 1070928 Ki = 18.6 nM T20401 COM2R4 1070933 Ki = 32.9 nM T20401 CKA4R5 1080680 Ki = 51 nM T20401 CDK1Z2 1085887 Ki > 50000 nM T20401 CA67JK 1124687 Ki = 49 nM T20401 CZ04BL 1136487 IC50 = 33.92 nM T20401 C4QX1Z 1146666 Ki = 9.3 nM T20401 CWD7G1 1147802 Ki = 660 nM T20401 CJ82NF 1178394 Ki = 14.5 nM T20401 C7A8VI 1211699 Ki > 1000 nM T20401 CYF34N 1211700 Ki > 1000 nM T20401 C7QP5E 1213792 Ki = 27 nM T20401 C6T0NU 1230924 Ki > 10000 nM T20401 C06ZSP 1234749 Ki = 132 nM T20401 C9IBF8 1241259 Ki = 3.6 nM T20401 CF1N3S 1277269 Ki = 36.1 nM T20401 CL87AM 1286568 Ki = 248 nM T20401 CA1I9S 1286583 Ki = 251 nM T20401 CE6W7O 1287222 Ki > 10000 nM T20401 CP60YD 1294363 Ki = 0.5 nM T20401 CYGO97 1300832 IC50 = 22.86 nM T20401 C5XNB4 1307068 Ki > 10000 nM T20401 C40CKN 1316238 Ki > 10000 nM T20401 CDWO53 1346695 Ki = 6.4 nM T20401 CC3G1N 1377410 Ki > 50000 nM T20401 C9DY2L 1488548 Ki = 650 nM T20401 CN5I0K 1505151 Ki = 38.1 nM T20401 CAHP42 1548275 Ki > 10000 nM T20401 CORY25 1581900 Ki = 340.94 nM T20401 C4YUX5 1594254 Ki = 330 nM T20401 C40YCV 1655994 Ki = 4 nM T20401 CU7KR6 1738244 Ki > 10000 nM T20401 C7XSO5 1748172 Ki > 10000 nM T20401 CGKP07 1748225 Ki > 10000 nM T20401 C98OLG 1775694 Ki > 10000 nM T20401 C5PU0O 1809247 IC50 = 27.16 nM T20401 CJ4G3B 1817956 Ki = 6.9 nM T20401 C9ZEH2 1825978 IC50 = 10.58 nM T20401 CY20OQ 1945421 Ki = 1.1 nM T20401 CTF8R5 1957305 Ki = 240 nM T20401 CR56WH 1968441 IC50 = 25.58 nM T20401 CK10DB 1977749 Ki = 75 nM T20401 C1DWG0 1989902 Ki = 3.8 nM T20401 CDQR23 2049187 Ki = 7.3 nM T20401 CP3RW6 2053748 Ki = 1.38 nM T20401 C2XA9Q 2054776 Ki = 5.012 nM T20401 C45WTO 2059531 Ki = 125 nM T20401 CSQJ97 2065546 Ki = 3455 nM T20401 CTK8C6 2089520 Ki = 47.6 nM T20401 C93VNU 2089779 Ki > 10000 nM T20401 C3W4PG 2192287 Ki = 4 nM T20401 C2O9YS 2196398 Ki = 4.9 nM T20401 C26OJZ 2206358 Ki = 18 nM T20401 CQS3A7 2207483 Ki > 10000 nM T20401 C3Y2CQ 2217668 Ki = 28 nM T20401 CO7JC2 2242987 Ki = 13 nM T20401 CH35BD 2265561 Ki = 16.98 nM T20401 C3FIK2 2268367 Ki = 133 nM T20401 CEW2Q3 2283723 Ki = 390 nM T20401 COB96D 2305168 Ki > 10000 nM T20401 C6FN0O 2316976 Ki = 73.6 nM T20401 CGW6L4 2318645 Ki = 3130 nM T20401 CD98QK 2333105 Ki > 10000 nM T20401 C1V0KL 2357187 Ki = 6.1 nM T20401 C3BJ4K 2368995 Ki = 474 nM T20401 CTJ42W 2368997 Ki = 374 nM T20401 C4TD8M 2388085 Ki = 3.1 nM T20401 C1TW9F 2457081 Ki > 10000 nM T20401 CJ10IX 2470552 Ki = 0.62 nM T20401 CR65UH 2471990 Ki > 50000 nM T20401 C95INQ 2476733 Ki = 2.4 nM T20401 C75SLD 2496330 Ki = 0.81 nM T20401 C2H4KT 2520594 Ki = 61 nM T20401 CBN52G 2566555 Ki = 28 nM T20401 CO1PU5 2570886 Ki = 26 nM T20401 CKH53Q 2723810 Ki = 24000000 nM T20401 C8YH7W 2733779 Ki > 100000 nM T20401 C0V7XB 2733782 Ki > 100000 nM T20401 C0W8UL 2735045 Ki = 305 nM T20401 CQ70UR 2755708 Ki = 1.9 nM T20401 CU60ZB 2755709 Ki = 1.7 nM T20401 CNG69U 2755712 Ki = 1.9 nM T20401 C58ISM 2755728 Ki = 8.1 nM T20401 C8QGL9 2760606 Ki > 10000 nM T20401 CNGK51 2781602 Ki = 28 nM T20401 CS0R6B 2789347 Ki > 10000 nM T20401 CD41AE 2795990 Ki = 74 nM T20401 CCOI52 2797418 Ki = 9829 nM T20401 C21FUI 2801263 Ki = 570 nM T20401 C4IDC5 2809317 Ki = 9000 nM T20401 C4V0MQ 2812911 Ki = 210 nM T20401 CPO6W3 2813478 Ki = 1150 nM T20401 CUI4Y8 2814914 Ki > 10000 nM T20401 CLFB40 2815883 Ki > 10000 nM T20401 C7A0CL 2826112 IC50 = 290 nM T20401 CDSN81 2826269 Ki = 0.23 nM T20401 CEY4J6 2858793 IC50 = 48.09 nM T20401 CU6D3W 2881615 IC50 > 10000 nM T20401 CBPO81 2882281 Ki = 12 nM T20401 CVA6F2 2893744 IC50 = 547 nM T20401 CE2GR3 2900806 Ki = 121000 nM T20401 CME74N 2904589 Ki = 220 nM T20401 CW9M7A 2952488 Ki = 40.9 nM T20401 CFO90D 2952737 Ki = 91 nM T20401 CQ9T8W 2970501 Ki = 10 nM T20401 C61OTP 2991092 Ki = 12 nM T20401 CZEH20 3003616 Ki = 81.5 nM T20401 CJ9LZ7 3051101 Ki > 100000 nM T20401 C6L2OC 3074858 Ki = 1.52 nM T20401 C87LCD 3082978 IC50 = 0.7 nM T20401 CN2Y5M 3083616 Ki > 100000 nM T20401 C9GT5Z 3083928 Ki > 100000 nM T20401 CY0OZ3 3090044 Ki = 8 nM T20401 C84TYH 3108089 IC50 = 3873 nM T20401 C49VDN 3132886 Ki > 10000 nM T20401 CQI7A2 3133127 Ki = 4.3 nM T20401 CP58HK 3344056 Ki = 20 nM T20401 C6V3ES 3365615 Ki = 0.9 nM T20401 CXU4J8 3377675 Ki = 7.9 nM T20401 C1K6IA 3379075 Ki = 9.3 nM T20401 C0FV7M 3414913 Ki = 16 nM T20401 CL6E2Y 3426384 Ki = 645.8 nM T20401 CT1NB8 3441996 Ki = 10.7 nM T20401 CZW71J 3476048 IC50 = 749.28 nM T20401 CP3BS4 3489403 Ki = 6 nM T20401 CHM17U 3496881 Ki = 2170 nM T20401 CIXH89 3516083 Ki = 6 nM T20401 C0VI6O 3524248 Ki > 50000 nM T20401 CM6R3S 3525535 Ki = 6 nM T20401 CKTY04 3538605 Ki = 27.5 nM T20401 C86GSL 3542746 Ki = 19 nM T20401 CHGS79 3551941 Ki = 95.6 nM T20401 CDI8T5 3576817 Ki = 27 nM T20401 C9L1HS 3586494 Ki = 2.2 nM T20401 CS5Z1Q 3614018 Ki = 142.5 nM T20401 CD0FL4 3627258 Ki = 12 nM T20401 CS4TM2 3638938 Ki = 24 nM T20401 CY89AI 3649509 Ki = 1160 nM T20401 C4WZG2 3657160 Ki = 39.1 nM T20401 CDY79J 3669864 Ki = 257000 nM T20401 CBED02 3683067 Ki = 119 nM T20401 C3REH6 3703019 IC50 = 8071 nM T20401 CQ5F9P 3724005 Ki = 23.1 nM T20401 CF9VG2 3770187 Ki = 590 nM T20401 CLW43B 3813634 Ki = 504 nM T20401 C2SY4L 3856570 Ki > 10000 nM T20401 CI3KT8 3936209 Ki > 10000 nM T20401 CV0KG3 3950536 Ki > 10000 nM T20401 CJ6D2S 3970972 Ki = 0.81 nM T20401 C8C4DV 4053995 Ki = 124 nM T20401 C5T1YZ 4056562 Ki = 230 nM T20401 C37VWB 4070422 Ki = 150 nM T20401 C25EPG 4073057 Ki = 5 nM T20401 C3CGU6 4094683 Ki = 24 nM T20401 CU2O1Y 4110011 Ki = 10900 nM T20401 C8DZ4B 4121769 Ki = 0.77 nM T20401 C9O0GV 4158561 Ki = 6.5 nM T20401 CPA56O 4180608 Ki = 17 nM T20401 CDNL69 4184455 Ki = 5000 nM T20401 CT57HM 4204917 Ki > 10000 nM T20401 CHOE81 4218706 Ki = 11 nM T20401 CORC17 4228388 Ki = 6 nM T20401 CD2P7T 4259683 Ki = 73 nM T20401 CV6BJ7 4262171 Ki > 40000 nM T20401 C2F9JP 4269754 Ki = 21 nM T20401 CUT26E 4274816 Ki > 50000 nM T20401 CUE97L 4276695 Ki > 10000 nM T20401 C5PM3E 4321567 Ki = 950000 nM T20401 CQ3P4I 4323207 Ki = 5 nM T20401 CI7UR5 4343483 Ki > 100000000 nM T20401 C37ZWJ 4369171 IC50 = 1.27 nM T20401 C0PX7R 4369172 IC50 = 1.15 nM T20401 CI6AE7 4377996 Ki = 9300 nM T20401 CQ2X7N 4389798 Ki = 2 nM T20401 C4E5VQ 4447263 Ki = 28.6 nM T20401 C96LCZ 4476238 Ki = 339 nM T20401 CIF43A 4572067 Ki = 12 nM T20401 CJ63TI 4578038 Ki = 0.88 nM T20401 CE5LO8 4578265 Ki = 741.7 nM T20401 C7RS2F 4583704 Ki > 1000 nM T20401 CAPM27 4598704 Ki > 50000 nM T20401 C3Q1WN 4607842 Ki = 33 nM T20401 CDK4L0 4608376 Ki = 570000 nM T20401 C02JOA 4616277 Ki = 600 nM T20401 CCP96V 4617978 Ki = 62 nM T20401 C6XVK9 4619076 Ki = 5329 nM T20401 CLSY09 4626049 Ki = 560 nM T20401 CLQ7U4 4627354 IC50 = 12.94 nM T20401 C3GDR0 4634582 Ki = 3500 nM T20401 CW1A4Z 4637857 Ki = 16 nM T20401 CPX3W6 4650747 Ki > 10000 nM T20401 CTM71V 4654716 Ki > 10000 nM T20401 CCB9Z5 4656684 Ki = 143 nM T20401 C2WI3U 4667972 Ki = 40 nM T20401 C07MRI 4712722 Ki = 600000 nM T20401 CWXE71 4718084 Ki = 8 nM T20401 C6RC3L 4718087 Ki = 4.6 nM T20401 C5FZ0L 4718107 IC50 = 153.18 nM T20401 CRL7B4 4718142 Ki = 4.2 nM T20401 CJM5F3 4718971 Ki = 12.7 nM T20401 CAG10X 4723337 IC50 = 670.72 nM T20401 C6B0OY 4723880 Ki = 10.7 nM T20401 C0MFT8 4801151 Ki > 10000 nM T20401 CSC7B8 4803242 Ki = 60.6 nM T20401 C7BIU4 4842634 IC50 = 21 nM T20401 CUA65R 4857564 Ki = 95.8 nM T20401 CX8C3P 4961927 Ki = 9.1 nM T20401 CX3RJ9 5005133 Ki = 337 nM T20401 CIP6Q8 5017140 Ki = 0.79 nM T20401 C7JBU0 5019114 Ki = 22.3 nM T20401 CF94ER 5032527 Ki > 10000 nM T20401 CD9V5J 5044227 Ki = 2600 nM T20401 C49FDN 5046067 Ki = 32.7 nM T20401 CTB04Y 5050031 Ki = 230 nM T20401 CX60DM 5067385 Ki = 24 nM T20401 C4OAL9 5070078 Ki = 4900 nM T20401 CN31CX 5071527 Ki = 46 nM T20401 CSG29M 5073140 Ki = 13 nM T20401 CP5F1Q 5100391 Ki = 5.18 nM T20401 CU8E4B 5133468 Ki > 100000 nM T20401 C7GXU1 5147921 Ki = 17500000 nM T20401 C89OCE 5155717 Ki = 12.4 nM T20401 CM9N8G 5161767 Ki > 10000 nM T20401 C6HM0R 5164092 Ki > 100000 nM T20401 C4HB1G 5172319 Ki = 1 nM T20401 CI8JY0 5172475 Ki = 19 nM T20401 CC37SW 5182516 Ki = 300 nM T20401 CZBY34 5220706 Ki = 13 nM T20401 CY9IV8 5223338 Ki = 10.2 nM T20401 CEN0L7 5227639 Ki = 11 nM T20401 CFQ62G 5232078 Ki > 100000 nM T20401 CF7G1E 5259801 IC50 = 3800 nM T20401 CEBD92 5272990 Ki = 61600 nM T20401 CP09FG 5272997 Ki = 23700 nM T20401 C4SV5T 5273568 Ki > 100000 nM T20401 CU4E5S 5273569 Ki = 94300 nM T20401 CZS0G5 5276565 IC50 > 10000 nM T20401 C3JN0F 5277465 IC50 > 10000 nM T20401 CRJK67 5277481 IC50 > 10000 nM T20401 CYF7S5 5277490 IC50 > 10000 nM T20401 CD1LZ7 5278580 Ki = 0.9 nM T20401 CNZ73E 5280567 Ki > 100000 nM T20401 CN10FM 5281793 Ki = 9594.4 nM T20401 CFB54A 5288859 Ki = 1.88 nM T20401 CA18OQ 5316302 Ki > 100000 nM T20401 CTJ01E 5317485 Ki > 100000 nM T20401 CI58XK 5319562 Ki = 800 nM T20401 CNO53D 5321265 Ki > 100000 nM T20401 C5Y6MA 5327300 Ki = 17 nM T20401 CP0R5H 5336569 Ki > 10000 nM T20401 C8PS4E 5358858 Ki > 100000 nM T20401 C4KHR2 5431473 IC50 = 33.13 nM T20401 CRVS37 5449904 Ki > 10000 nM T20401 C2UN6J 5462815 Ki = 570000 nM T20401 CH5OM1 5463917 Ki = 11600000 nM T20401 CG76KE 5470394 Ki = 0.6 nM T20401 CXEW32 5491996 Ki > 100000 nM T20401 C7RG3L 5496307 Ki = 4300 nM T20401 CX71JE 5682293 Ki > 10000 nM T20401 CWYU91 5742696 Ki = 2650 nM T20401 CU0FW5 5743063 Ki = 1930 nM T20401 C4VZP8 5765787 Ki = 5.4 nM T20401 CWL5R2 5765789 Ki = 6 nM T20401 CK0M4A 5910585 Ki > 100000 nM T20401 C7T1DV 5956379 Ki = 0.6 nM T20401 C01AGL 6097189 Ki = 1870000 nM T20401 CHJ3V8 6102658 Ki = 310 nM T20401 CJZ47Y 6365232 Ki = 86000 nM T20401 CPVB19 6399220 Ki = 89000000 nM T20401 CMD1Q0 6460079 Ki = 1.8 nM T20401 CS4KQ6 6482974 Ki = 9650 nM T20401 C9L8AX 6537802 Ki > 200000 nM T20401 C91GBW 6604453 Ki = 15.3 nM T20401 C65FRB 6852128 Ki = 12 nM T20401 CPFV65 6916013 Ki = 39 nM T20401 CK85ZF 7022526 IC50 > 50000 nM T20401 C0W5GD 7130726 Ki = 2.3 nM T20401 CWL9C2 7382212 Ki > 10000 nM T20401 C75SBG 7382231 Ki > 50000 nM T20401 C6U9MT 7382238 Ki = 43.5 nM T20401 CY57CX 7382249 Ki > 10000 nM T20401 C5TK0N 7463363 IC50 = 9430 nM T20401 C7RM6F 7463364 IC50 = 8660 nM T20401 C9UJB7 7463369 IC50 = 6510 nM T20401 CKCM96 7463376 Ki = 910 nM T20401 CDCP43 7766335 Ki > 50000 nM T20401 CTH8D3 7785988 Ki > 10000 nM T20401 C95AKP 7794397 Ki > 10000 nM T20401 C6S5HK 7832430 Ki > 10000 nM T20401 C1EKW8 7996519 Ki > 40000 nM T20401 C6WG0N 8007128 Ki = 30 nM T20401 C67SFK 8084575 Ki = 86.8 nM T20401 CQ0Z4E 8098235 Ki = 89 nM T20401 CCW8R6 8190912 Ki = 203 nM T20401 CSW01Z 8272034 Ki > 10000 nM T20401 C9BAM4 8281641 Ki = 7.5 nM T20401 C3WQ9M 8866559 Ki = 38.2 nM T20401 C5CS1Y 9314410 Ki = 3.8 nM T20401 C3SA2N 9314413 Ki = 0.63 nM T20401 C47VSJ 9572721 Ki > 10000 nM T20401 CIJ25V 9794947 IC50 = 8000 nM T20401 CY42UH 9812913 Ki = 950000 nM T20401 C7SRM4 9837496 IC50 = 8810 nM T20401 C0EJ1Q 9847197 Ki = 1.4 nM T20401 C47IMW 9863339 Ki = 0.14 nM T20401 CT37DQ 9879717 Ki = 0.69 nM T20401 C54XWL 9898889 Ki = 950000 nM T20401 C6LAR2 9942169 Ki = 260000 nM T20401 C6YW0Q 9942868 Ki = 200.5 nM T20401 CSIY73 9952009 IC50 > 100000 nM T20401 CYP7E9 9964347 Ki = 270000 nM T20401 C24ZVR 9982838 Ki = 4.14 nM T20401 CJS4I3 9990000 Ki = 3.4 nM T20401 CIN68V 9998184 Ki = 84 nM T20401 CY47OI 9998322 Ki = 30 nM T20401 C6TO0A 10001582 Ki = 36 nM T20401 CXD28H 10015065 Ki = 1.5 nM T20401 CQ79OY 10015713 Ki = 125025903 nM T20401 CNKD31 10016330 Ki = 526.9 nM T20401 C4UEV9 10016475 Ki > 10000 nM T20401 CF6RN0 10018880 Ki = 106 nM T20401 CX4MK5 10019750 Ki = 35 nM T20401 CGU6P4 10021113 IC50 = 1.28 nM T20401 CKOV96 10023066 Ki = 6 nM T20401 CQL10G 10026448 Ki = 2 nM T20401 C6DGR7 10027203 Ki > 200 nM T20401 CX2W9O 10037048 IC50 = 8850 nM T20401 CY2SP7 10037665 IC50 = 626 nM T20401 C7L0EZ 10038370 IC50 = 590 nM T20401 CZHE98 10038620 IC50 = 6.8 nM T20401 CPDC51 10040931 Ki = 47.5 nM T20401 CO39PK 10042482 Ki = 8 nM T20401 CI5AR1 10044828 Ki = 7 nM T20401 C1H9KF 10046686 Ki = 1.43 nM T20401 C5Q1FI 10052644 Ki = 2 nM T20401 C5X7GY 10059582 Ki = 2192 nM T20401 CWM01R 10059806 Ki = 5636 nM T20401 CXQV82 10061571 IC50 = 2.46 nM T20401 COWD07 10062976 Ki = 5 nM T20401 C69DPZ 10068042 IC50 > 100000 nM T20401 C70CWE 10068417 IC50 = 0.58 nM T20401 C6FKM3 10069411 Ki = 10 nM T20401 CY8F0E 10076040 Ki > 100000 nM T20401 CU7DJ1 10081163 Ki = 70 nM T20401 C0P5XV 10081897 Ki = 871.7 nM T20401 CD58EL 10083644 Ki > 50000 nM T20401 CXJ03P 10086394 IC50 = 4.7 nM T20401 CCR24T 10087045 Ki = 42 nM T20401 CZU5A2 10088969 Ki = 6 nM T20401 C2AGT9 10090122 IC50 = 4.6 nM T20401 CHUS78 10090395 IC50 = 2.9 nM T20401 CTE08N 10091688 IC50 = 18 nM T20401 CT64MX 10094466 Ki = 250034536.2 nM T20401 CRN29P 10104483 Ki = 1.1 nM T20401 C4ENU8 10107524 IC50 = 160 nM T20401 C7WU0A 10107532 Ki = 2362 nM T20401 CAQ6I1 10131078 Ki = 7.5 nM T20401 CXD91O 10136406 Ki = 5.2 nM T20401 CVRZ27 10198038 IC50 = 7410 nM T20401 C63AZQ 10198750 Ki = 7.4 nM T20401 CUR4O7 10198795 Ki = 8.8 nM T20401 CJV68L 10220266 Ki = 685.5 nM T20401 CM4E8G 10243877 Ki = 2 nM T20401 C4E1JQ 10245883 Ki = 50 nM T20401 C4YQG0 10255391 IC50 = 2.18 nM T20401 CX50AK 10266719 Ki = 240 nM T20401 CC9XT4 10267015 Ki = 12 nM T20401 CLM6Z5 10290835 Ki > 10000 nM T20401 CS3CE7 10313432 Ki = 13 nM T20401 CHEN62 10316843 Ki = 3.32 nM T20401 C74DMN 10316844 IC50 = 5 nM T20401 CZ72IC 10318089 Ki = 4 nM T20401 CQ8A0I 10328097 Ki = 6863.3 nM T20401 CN40WD 10331524 Ki = 1141 nM T20401 CTL91E 10333887 IC50 = 3.18 nM T20401 CU9OI5 10334780 Ki = 20 nM T20401 CEKT36 10335685 Ki = 1.19 nM T20401 CUE81P 10337354 Ki > 10000 nM T20401 CRHU49 10338639 Ki = 8 nM T20401 CKI9O5 10342490 Ki = 0.97 nM T20401 CX6P1I 10358994 Ki = 10 nM T20401 CH4I9P 10360342 Ki = 10 nM T20401 CR4FJ3 10361377 IC50 = 200 nM T20401 C58IYR 10366827 Ki = 560 nM T20401 CYC32P 10367512 IC50 = 1.45 nM T20401 C3HBY6 10375558 Ki = 50 nM T20401 CP0EX9 10379035 Ki = 2.9 nM T20401 CT9VJ3 10383097 Ki = 16 nM T20401 C1O2FH 10383098 Ki = 21 nM T20401 CSU78V 10384414 IC50 = 7 nM T20401 CP2XW6 10387325 Ki = 10 nM T20401 CUS1B8 10399861 IC50 = 12.8 nM T20401 C0S4RA 10400708 Ki = 18 nM T20401 CVW18K 10409391 Ki = 1 nM T20401 C5IK7H 10420920 Ki = 1.5 nM T20401 C4MI8O 10423003 Ki = 10 nM T20401 C87TXN 10423541 IC50 = 5 nM T20401 C07JML 10423646 IC50 = 13 nM T20401 CI60TB 10423771 Ki = 10 nM T20401 CFGK83 10430595 Ki = 0.7 nM T20401 CVIN94 10439991 Ki = 8790.2 nM T20401 CIC54M 10452478 Ki = 24 nM T20401 C6T8VC 10456675 Ki = 107 nM T20401 CD80XW 10465553 IC50 = 16 nM T20401 CED61Q 10467688 Ki = 85 nM T20401 C6TYP0 10467861 Ki > 10000 nM T20401 C25NJB 10471772 Ki = 420 nM T20401 CM4B5L 10473220 IC50 = 13 nM T20401 C13JVK 10477954 Ki = 15 nM T20401 CA3CV1 10492408 Ki = 13696197.19 nM T20401 CEV92X 10493372 Ki = 111 nM T20401 C41KHC 10494655 Ki = 11 nM T20401 CJFC96 10495006 Ki = 4 nM T20401 C4ZV9X 10495711 Ki = 11 nM T20401 C3Y0AX 10497272 Ki = 8 nM T20401 CE2XQ6 10497552 Ki = 9 nM T20401 CPMT67 10497717 Ki = 5 nM T20401 CSZ1K0 10499069 Ki = 3 nM T20401 CL8O6I 10500340 Ki = 16 nM T20401 CVID65 10500886 Ki > 200 nM T20401 CBL23S 10502993 Ki = 9 nM T20401 CV0FT4 10503780 Ki = 19 nM T20401 CA95ZO 10504238 Ki = 36 nM T20401 CU8E4S 10505384 Ki = 50 nM T20401 CRS2V1 10505991 Ki = 400 nM T20401 CRJ8O1 10506509 Ki = 7 nM T20401 CH6A2O 10507009 Ki = 270 nM T20401 C3TCR7 10507836 Ki = 21 nM T20401 CRNO69 10508249 Ki = 6 nM T20401 CR3AL4 10508270 Ki = 107 nM T20401 CG0MZ8 10508351 Ki = 6 nM T20401 C52EMX 10509011 Ki = 22 nM T20401 CIW1L8 10509163 Ki = 2 nM T20401 C3G4PQ 10509380 Ki = 72 nM T20401 CD41CA 10512636 Ki = 96.5 nM T20401 CJZ67W 10515762 Ki = 9 nM T20401 CM62BT 10516272 Ki = 31253596.44 nM T20401 C4SQ5V 10517256 Ki = 33334964.73 nM T20401 CR63LA 10518811 Ki = 6 nM T20401 C48KTA 10519415 Ki = 18518252.44 nM T20401 CFOE60 10519650 Ki = 14800 nM T20401 CM0K8P 10519868 Ki = 3 nM T20401 CXD8I5 10523292 Ki = 15 nM T20401 CZT6S0 10523695 Ki = 15 nM T20401 CU2E3A 10524550 Ki = 2 nM T20401 CZ4LU8 10524990 Ki = 9 nM T20401 CQL8S4 10525380 Ki = 1.5 nM T20401 C7UY4Z 10526065 Ki = 11 nM T20401 CM4Q7C 10526660 Ki = 35 nM T20401 CUJI62 10527611 Ki = 430 nM T20401 C7Z1LE 10527692 Ki = 250 nM T20401 CK43UF 10528302 Ki = 460 nM T20401 CG1M8V 10529267 Ki = 215 nM T20401 CGK37L 10529602 Ki = 118 nM T20401 CI6SU7 10530110 Ki = 34 nM T20401 CTP62O 10530164 Ki = 19 nM T20401 CU6HX8 10530223 Ki = 103 nM T20401 C6C7YQ 10531119 Ki = 544 nM T20401 CA5C0S 10531121 Ki = 275 nM T20401 CND17Q 10532205 Ki = 10 nM T20401 C3PO6V 10532224 Ki = 16 nM T20401 CC0EB5 10532491 Ki = 13 nM T20401 CU6YM4 10532987 Ki = 680 nM T20401 CJ1D2U 10533054 Ki = 70 nM T20401 CWQY26 10535227 Ki > 10000 nM T20401 CT04WN 10537366 Ki = 210 nM T20401 C5PMH4 10539133 Ki = 193 nM T20401 C5G8EX 10540518 Ki = 28 nM T20401 C5I3JC 10541189 Ki = 121 nM T20401 C9EM7W 10543041 Ki = 8 nM T20401 CF72EQ 10543283 Ki = 199986187 nM T20401 C3KHS0 10543744 Ki = 10 nM T20401 C81ZYH 10543818 Ki = 23 nM T20401 C5S9PM 10546426 Ki = 4 nM T20401 CIN60X 10548978 Ki = 2 nM T20401 C0S7OI 10549020 Ki = 125 nM T20401 C5JS8L 10549329 Ki > 200 nM T20401 CY93AQ 10549606 Ki = 40 nM T20401 CN8KT4 10550727 Ki = 13 nM T20401 CW1L5G 10550795 Ki = 250034536.2 nM T20401 C3ALP8 10550907 Ki = 110 nM T20401 CCTN57 10551138 Ki = 10 nM T20401 CQ2U6H 10552761 Ki = 0.4 nM T20401 C31INC 10553159 Ki = 230 nM T20401 C8CJ3W 10554523 Ki = 220 nM T20401 C9CHQ8 10554752 Ki = 46 nM T20401 C4C5YD 10555371 Ki = 11 nM T20401 CDJ9O6 10555708 Ki = 8 nM T20401 C6QH5Y 10555828 Ki = 66 nM T20401 CJ74IY 10556211 Ki = 25 nM T20401 CVJ85T 10556224 Ki = 8 nM T20401 CV79UJ 10556471 Ki = 12 nM T20401 CUM09Y 10563097 Ki = 8926886.23 nM T20401 C08EWG 10563541 Ki = 41 nM T20401 CMXB05 10564634 Ki = 100000000 nM T20401 CQP6G1 10565056 Ki = 187 nM T20401 CY79EX 10565133 Ki = 15149559.32 nM T20401 CCKE29 10566405 Ki = 20450 nM T20401 C7UYX1 10566734 Ki = 7 nM T20401 C7U2DR 10567673 Ki = 27 nM T20401 CLFN25 10567759 Ki = 121 nM T20401 C3W9QA 10568362 Ki = 25 nM T20401 CD8T0J 10568499 Ki = 5 nM T20401 CT6BA5 10572515 Ki = 40 nM T20401 C8RD4P 10573046 Ki = 30 nM T20401 CRUW05 10573729 Ki = 76913044.03 nM T20401 CP71JY 10573928 Ki = 15 nM T20401 CRO7J0 10574278 Ki = 0.5 nM T20401 C2PH8Q 10575017 Ki = 6 nM T20401 C9N8YQ 10575994 Ki = 2 nM T20401 CQ3XL8 10576231 Ki = 0.7 nM T20401 C8CMG3 10577063 Ki = 8 nM T20401 CF3A4I 10577600 Ki = 61 nM T20401 CN8R3Y 10577727 Ki = 38 nM T20401 CQV65S 10578334 Ki = 51 nM T20401 C6CNQ7 10578619 Ki = 32 nM T20401 CCNW04 10578621 Ki = 275 nM T20401 C6HO9B 10578774 Ki = 9 nM T20401 C8I9FB 10580194 Ki = 2 nM T20401 C28OGL 10580382 Ki = 3 nM T20401 C8UW9L 10580477 Ki = 550 nM T20401 C9CF5Q 10580554 Ki = 2 nM T20401 CJ8IW3 10581021 Ki = 32 nM T20401 CAVB38 10586310 Ki = 180 nM T20401 C73KXU 10586607 Ki = 24600 nM T20401 C0BPD3 10589291 Ki = 9 nM T20401 CD4V5G 10590334 Ki = 5 nM T20401 C0N1IM 10590553 Ki = 12 nM T20401 C6KD1Z 10591288 Ki = 30 nM T20401 C8J6HS 10591505 Ki = 5 nM T20401 CB20LM 10594000 Ki = 120 nM T20401 C25DOL 10594934 Ki = 2 nM T20401 CBM48L 10596042 Ki = 31 nM T20401 CAZ36G 10596413 Ki = 1.5 nM T20401 C1JRL7 10597208 Ki = 10 nM T20401 CH37KM 10599305 Ki = 10 nM T20401 C3VZX6 10599546 Ki = 43 nM T20401 CAL87S 10599609 Ki = 79 nM T20401 CH6J5O 10600355 Ki = 21 nM T20401 CY8HT7 10601085 Ki = 425 nM T20401 C8LE1Z 10601296 Ki = 11 nM T20401 CO8D2C 10602116 Ki = 21 nM T20401 CM6I8S 10602258 Ki = 8 nM T20401 CWG1C7 10602601 Ki = 7 nM T20401 CZB76C 10602667 Ki = 20 nM T20401 CP4AY9 10603234 Ki = 13 nM T20401 C9SLH3 10603241 Ki = 4 nM T20401 C9YR2K 10603335 Ki = 19 nM T20401 CJNP46 10603338 Ki = 70 nM T20401 C6G0ZI 10603469 Ki = 15 nM T20401 C6C9ZB 10603761 Ki = 20 nM T20401 CT4EC1 10603881 Ki = 69 nM T20401 C73UOS 10604129 Ki = 15 nM T20401 C65GKZ 10609913 Ki = 9 nM T20401 C5G9MI 10610114 Ki = 1.1 nM T20401 CZS6O0 10610757 Ki = 6 nM T20401 CN38WB 10611730 Ki = 6 nM T20401 C8N4EO 10614528 Ki = 105 nM T20401 C2PRM1 10615166 Ki = 35 nM T20401 CM46AO 10615795 Ki = 500 nM T20401 C78TRD 10617314 Ki = 10 nM T20401 C1EIP0 10618881 Ki = 35 nM T20401 CK92EO 10619964 Ki = 37033946.94 nM T20401 CF85VP 10620016 Ki = 15 nM T20401 CSY79P 10620807 Ki = 25 nM T20401 CV08XY 10621281 Ki = 100000000 nM T20401 CU61LT 10621497 Ki = 166686335.9 nM T20401 CM9H5A 10623288 Ki = 31 nM T20401 C8HRI3 10623948 Ki = 78 nM T20401 C97JCY 10625036 Ki = 120 nM T20401 CU3YT8 10625038 Ki = 9 nM T20401 CVN72J 10625060 Ki = 110 nM T20401 C4FLA9 10625484 Ki = 90 nM T20401 CGI03J 10625651 Ki = 420 nM T20401 CMQC23 10625732 Ki = 6 nM T20401 CGB5S0 10626619 Ki = 350 nM T20401 CCX2K6 10627219 Ki = 16 nM T20401 CWN3O4 10628503 Ki = 15 nM T20401 C9N2ZH 10629041 Ki = 755 nM T20401 CFL47V 10629052 Ki = 1.5 nM T20401 C9TSQ6 10632698 Ki = 3800 nM T20401 C4I2QF 10633163 Ki = 124 nM T20401 C2OHP3 10635833 Ki = 32 nM T20401 C0KA3F 10637879 Ki = 30 nM T20401 C7YOD1 10637941 Ki = 190 nM T20401 C4VQC3 10638194 Ki = 18700 nM T20401 CN8IR0 10638758 Ki = 350 nM T20401 CU6IE1 10640069 Ki = 6 nM T20401 CPH72T 10640797 Ki = 730 nM T20401 CN6HA4 10642039 Ki = 9 nM T20401 C2ULM5 10642205 Ki = 250034536.2 nM T20401 CJV5L1 10643532 Ki = 23 nM T20401 CC8T9S 10645605 Ki = 9 nM T20401 CNAE38 10647590 Ki = 0.2 nM T20401 CIW58E 10648512 Ki = 385 nM T20401 C9V3WZ 10649387 Ki = 0.5 nM T20401 CCI16T 10649726 Ki = 125 nM T20401 CK2F6I 10649728 Ki = 240 nM T20401 CQB3T1 10650115 Ki = 0.26 nM T20401 CG4HL1 10650150 Ki = 16 nM T20401 CZN6S5 10650429 Ki = 0.7 nM T20401 CC4UM6 10650450 Ki = 321 nM T20401 CW2AC6 10651479 Ki = 2 nM T20401 CZ9GS7 10651537 Ki = 21 nM T20401 CSV84J 10651858 Ki = 9 nM T20401 CFJA05 10651893 Ki = 67 nM T20401 CE14NG 10652046 Ki = 540 nM T20401 CZHL98 10658802 Ki = 5069907.08 nM T20401 CE24FZ 10660854 Ki = 200 nM T20401 CIMZ90 10663338 Ki = 275 nM T20401 C19DBM 10663960 Ki = 9 nM T20401 C4SX7R 10665257 Ki = 15 nM T20401 C6VBM9 10665468 Ki = 7 nM T20401 C09FLT 10665545 Ki = 90907559.74 nM T20401 CMN37R 10666283 Ki = 0.9 nM T20401 CC8WH4 10666501 Ki = 36 nM T20401 C3E0ZP 10667414 Ki = 21 nM T20401 C9IL3M 10670278 Ki = 15 nM T20401 C1W7CO 10671070 Ki = 80 nM T20401 CB39ZS 10671185 Ki = 320 nM T20401 CWB19K 10671441 Ki = 74 nM T20401 CWQ58H 10671476 Ki = 8 nM T20401 CB6CA9 10672102 Ki = 98 nM T20401 CQK8V3 10673297 Ki = 230 nM T20401 CVX50Z 10673405 Ki = 5 nM T20401 CJ9D7F 10673563 Ki = 36 nM T20401 C6AH3Z 10673625 Ki = 30 nM T20401 CETF96 10673746 Ki = 440 nM T20401 C79OXJ 10673953 Ki = 39 nM T20401 CY9W0O 10674571 Ki = 18 nM T20401 C02FIM 10674633 Ki = 8 nM T20401 CL6GZ4 10675046 Ki = 4 nM T20401 CR2D8E 10675795 Ki = 96 nM T20401 C6B8JA 10675931 Ki = 60 nM T20401 CSZ39G 10676062 Ki = 440 nM T20401 CS2FT7 10676818 Ki = 98 nM T20401 CA18CD 10680096 IC50 = 5.2 nM T20401 CN1ZW0 10682584 Ki = 5495408.74 nM T20401 C9IAB0 10685830 Ki = 280 nM T20401 C2UH7Z 10687216 Ki = 242 nM T20401 CGJ7L6 10691042 Ki = 3 nM T20401 CVHO36 10692638 Ki = 100 nM T20401 C4BQK5 10693598 Ki = 0.6 nM T20401 C17ICZ 10693904 Ki = 1300 nM T20401 C0TOK2 10695275 Ki = 0.3 nM T20401 CHG04R 10695589 Ki = 150 nM T20401 CH63NB 10695632 Ki = 180 nM T20401 C2YH7O 10696741 Ki = 210 nM T20401 CRL2U7 10696743 Ki = 493 nM T20401 CE82AF 10697359 Ki = 42 nM T20401 CV2RJ5 10697379 Ki = 205 nM T20401 C0VF5D 10697562 Ki = 485 nM T20401 CT59ZG 10697685 Ki = 290 nM T20401 C0NM4D 10698231 Ki = 71 nM T20401 C6MG9R 10698477 Ki = 6 nM T20401 C1P2SH 10698664 Ki = 419 nM T20401 CKV21F 10699169 Ki = 5 nM T20401 C62VLP 10699783 Ki = 5 nM T20401 CXZ97V 10699991 Ki = 0.6 nM T20401 C0DIN6 10700505 Ki = 2 nM T20401 C5WSA3 10704587 Ki = 200 nM T20401 C5E8QF 10707457 Ki = 35 nM T20401 C59QWT 10708731 Ki = 32255219.38 nM T20401 CFZ65M 10710739 Ki = 5100 nM T20401 C8NH6B 10711889 Ki = 270 nM T20401 C6D2TJ 10712038 Ki = 2135 nM T20401 CE8L3N 10712383 Ki = 7 nM T20401 C9LD0S 10712555 Ki = 4 nM T20401 CLV42Z 10713226 Ki = 25 nM T20401 CRI51E 10713868 Ki = 1600 nM T20401 C9PXS4 10714881 Ki = 6 nM T20401 CGNP20 10715470 Ki = 14 nM T20401 C23LAY 10715903 Ki = 7 nM T20401 C7JS2I 10716079 Ki = 10 nM T20401 CX8YI4 10716240 Ki = 30 nM T20401 CI6Y4G 10716883 Ki = 90 nM T20401 C3TGW8 10717400 Ki = 18 nM T20401 CG3NP5 10718314 Ki = 1.1 nM T20401 CDV6R8 10718340 Ki = 2 nM T20401 CS9X0E 10719552 Ki = 5 nM T20401 CSJ14E 10720061 Ki = 200 nM T20401 C1L8UA 10720537 Ki = 0.5 nM T20401 C8WJK7 10721281 Ki = 7 nM T20401 CB59QH 10721415 Ki = 235 nM T20401 CT87NP 10721547 Ki = 8 nM T20401 CNF6H0 10721639 Ki = 510 nM T20401 CT65DL 10722417 Ki = 8 nM T20401 C2OYQ1 10722508 Ki = 15 nM T20401 C3K1DN 10722521 Ki = 103 nM T20401 C4VOP2 10722619 Ki = 5 nM T20401 C42TPS 10722680 Ki = 36 nM T20401 CSE58B 10723137 Ki = 14 nM T20401 CV9A8J 10723227 Ki = 54 nM T20401 C4GX0Y 10723329 Ki = 10 nM T20401 CR0M8G 10723505 Ki = 0.5 nM T20401 C2A6LI 10728925 Ki = 187 nM T20401 CR5U3C 10734581 Ki = 30 nM T20401 CGX10J 10736890 Ki = 45 nM T20401 C2ZLE4 10737428 Ki = 7.5 nM T20401 C5G2OP 10737443 Ki = 4 nM T20401 C83KNR 10737789 Ki = 36 nM T20401 CU9YA6 10737942 Ki = 111096403.5 nM T20401 CL5U3V 10738713 Ki = 1040 nM T20401 CGH3P0 10738795 Ki = 12 nM T20401 CGTX61 10738796 Ki = 13 nM T20401 C8Z9IL 10739376 Ki = 17 nM T20401 CNW7S5 10740344 Ki = 33 nM T20401 CD3HN0 10740410 Ki = 71433182.62 nM T20401 C4FWC9 10740485 Ki = 15 nM T20401 CB9T4M 10742338 Ki = 160 nM T20401 CN30YJ 10742576 Ki = 21 nM T20401 CBF1Z5 10742874 Ki = 3 nM T20401 CEBQ21 10744110 Ki = 0.5 nM T20401 CCRG49 10744718 Ki = 150 nM T20401 C6O7PQ 10744771 Ki = 10 nM T20401 CW6Q1M 10744854 Ki = 3 nM T20401 C7WHI1 10745371 Ki = 595 nM T20401 CG4OI8 10745793 Ki = 35 nM T20401 C0KN7Z 10745795 Ki = 650 nM T20401 C6IP0J 10746098 Ki = 6 nM T20401 CTG8L5 10746646 Ki = 51 nM T20401 CLMA04 10747000 Ki = 110 nM T20401 CG8K9X 10747080 Ki = 37 nM T20401 CG1MT4 10747258 Ki = 69 nM T20401 C0OC6N 10747270 Ki = 17 nM T20401 CXE89A 10747447 Ki = 2 nM T20401 C7BSK4 10747629 Ki = 20 nM T20401 C8DL1Z 10747766 Ki = 11 nM T20401 CY1WX7 10747964 Ki = 12 nM T20401 CB6M3O 10747965 Ki = 21 nM T20401 CLN70E 10750432 IC50 = 8 nM T20401 C7MEP5 10752797 Ki = 250 nM T20401 CRG5Z7 10753241 Ki = 10 nM T20401 CO8B6L 10756624 Ki = 36 nM T20401 CA3F1N 10758013 Ki = 8 nM T20401 CQUP90 10759040 Ki = 550 nM T20401 C14QMV 10759047 Ki = 150 nM T20401 CY4RA2 10759222 Ki = 36 nM T20401 CA5BQ1 10763396 Ki = 8 nM T20401 CBHI21 10763843 Ki = 1 nM T20401 C3HVQ9 10764510 Ki = 50 nM T20401 CTK7W3 10765251 Ki = 145 nM T20401 CZ8S0A 10765253 Ki = 250 nM T20401 CR4J2Z 10765565 Ki = 8 nM T20401 C4R2FB 10765728 Ki = 156 nM T20401 C0XNP9 10765735 Ki = 2 nM T20401 CXD7E4 10765823 Ki = 10 nM T20401 CH78WD 10766083 Ki = 20 nM T20401 CF5I7H 10766126 Ki = 170 nM T20401 C69MAB 10766339 Ki = 23 nM T20401 CA6C0Z 10766622 Ki = 56 nM T20401 CIB3E5 10766650 Ki = 60 nM T20401 C06MYS 10766652 Ki = 8 nM T20401 CVD0H3 10766865 Ki = 5 nM T20401 C96BYJ 10767057 Ki = 12 nM T20401 C2K3XN 10767400 Ki = 9 nM T20401 CM8JR1 10767828 Ki = 5 nM T20401 C9Z3EL 10767989 Ki = 31 nM T20401 CRS6F0 10768100 Ki = 7 nM T20401 C7X3PW 10768529 Ki = 580 nM T20401 C3L4OV 10768593 Ki = 7 nM T20401 CHVB87 10768870 Ki = 370 nM T20401 CMS9R1 10769153 Ki = 8 nM T20401 C4CT1D 10769199 Ki = 49 nM T20401 CQ15VI 10769549 Ki = 1.5 nM T20401 CZDJ14 10770028 Ki = 12 nM T20401 C06DZW 10770030 Ki = 15 nM T20401 CD4VK5 10770656 Ki = 3 nM T20401 CDU8X0 10770816 Ki = 11 nM T20401 CHQ83W 10778778 Ki = 100000000 nM T20401 CYG79W 10779489 Ki = 160 nM T20401 C1T9VB 10782719 Ki = 9 nM T20401 C31CQW 10783063 Ki = 33334964.73 nM T20401 C40YHF 10783082 Ki = 19 nM T20401 CRXH95 10784749 Ki = 9 nM T20401 C7T1ZF 10788101 Ki = 40 nM T20401 C3P7LZ 10792025 Ki = 116 nM T20401 CDO17N 10792606 Ki = 620 nM T20401 C5Q0HP 10792608 Ki = 390 nM T20401 CCF8T2 10792692 Ki = 19 nM T20401 CMY20D 10792820 Ki = 5 nM T20401 CR9A3S 10792923 Ki = 15 nM T20401 CCYS21 10793062 Ki = 1 nM T20401 CK5ZL2 10793077 Ki = 42 nM T20401 CHD5Q2 10793387 Ki = 18 nM T20401 CX0BW6 10793389 Ki = 7 nM T20401 CEY35S 10793458 Ki = 17 nM T20401 CFL4G8 10800492 Ki = 12 nM T20401 CH1F0I 10803110 Ki = 200 nM T20401 C25VZF 10804238 Ki = 245 nM T20401 CU1BS8 10804376 Ki = 250 nM T20401 CGY6S7 10804696 Ki = 38 nM T20401 C7N2LO 10805708 Ki = 260 nM T20401 C1QF3B 10806893 Ki = 44 nM T20401 CH1A4N 10807238 Ki = 4 nM T20401 CC0V8S 10808608 Ki = 0.9 nM T20401 CU9F7V 10810684 Ki = 170 nM T20401 CJGV81 10810883 Ki = 9 nM T20401 C58LOZ 10812489 Ki = 33 nM T20401 C42JTI 10813047 Ki = 10 nM T20401 CQR74O 10813858 Ki = 20 nM T20401 C4Q1BT 10814610 Ki = 125 nM T20401 CPG8X7 10815580 Ki = 38 nM T20401 CIU0T4 10815639 Ki = 45 nM T20401 C9S1KI 10816020 Ki = 314 nM T20401 CZ8SC0 10816485 Ki = 15 nM T20401 CDX47C 10817418 Ki = 51 nM T20401 CPU04C 10817804 Ki = 4 nM T20401 CI21MQ 10817828 Ki = 550 nM T20401 CW4J0M 10817935 Ki = 12 nM T20401 CR6WQ9 10818727 Ki = 35 nM T20401 CQBR40 10825041 Ki = 33 nM T20401 CVN37O 10825297 Ki = 10 nM T20401 CW9YL5 10827620 Ki = 6 nM T20401 CIW28L 10829558 Ki = 36 nM T20401 C36NTE 10829886 Ki = 200 nM T20401 CHE35M 10832570 Ki = 29 nM T20401 C3TN8I 10832697 Ki = 19 nM T20401 CA13RM 10833200 Ki = 2 nM T20401 COE82D 10833334 Ki = 11 nM T20401 CQM97L 10833411 Ki = 13 nM T20401 CMI8K1 10833817 Ki = 13 nM T20401 C9M1JI 10834357 Ki > 200 nM T20401 C6U5RE 10834502 Ki = 50 nM T20401 C1R4OZ 10836567 Ki = 12 nM T20401 CWF8K2 10836730 Ki = 2 nM T20401 CLS5J3 10836786 Ki = 60 nM T20401 C0IY7D 10836837 Ki = 8 nM T20401 C3NIE1 10836973 Ki = 3 nM T20401 CO6C3T 10837292 Ki = 12 nM T20401 CR0E9Q 10837740 Ki = 85 nM T20401 C3XU6W 10838049 Ki = 10 nM T20401 C32QME 10838459 Ki = 21 nM T20401 C2P7QW 10839526 Ki = 12 nM T20401 CBE3L7 10839725 Ki = 18 nM T20401 CLIK46 10840741 Ki = 300 nM T20401 CM4ZJ7 10841903 Ki = 55 nM T20401 CX9B7K 10841917 Ki = 410 nM T20401 CJI5F0 10841980 Ki = 55 nM T20401 CWVN58 10842131 Ki = 18 nM T20401 CG6XO9 10842189 Ki = 125 nM T20401 CMA41F 10842208 Ki = 1 nM T20401 C93MDS 10842492 Ki = 15 nM T20401 C98LNY 10842547 Ki = 5 nM T20401 C5Z3AD 10842801 Ki = 0.6 nM T20401 C3W8OJ 10842917 Ki = 16 nM T20401 CW28MA 10843175 Ki = 3 nM T20401 CB2KJ7 10847811 Ki = 40 nM T20401 CO2SP9 10847812 Ki = 115 nM T20401 CQ0HY2 10848746 Ki = 39 nM T20401 C0ZQ7X 10849797 Ki = 4716284.55 nM T20401 CMH6X5 10850981 Ki = 20 nM T20401 C06ORC 10851952 Ki = 10 nM T20401 C98OIB 10852025 Ki = 11 nM T20401 CH0A6S 10852944 Ki = 42 nM T20401 CLQ6M8 10854347 Ki = 199986187 nM T20401 CF9SV4 10861185 Ki = 7 nM T20401 CZ4P8F 10862789 Ki = 43 nM T20401 C1B2IY 10863970 Ki = 0.8 nM T20401 C19MNG 10864178 Ki = 280 nM T20401 CPN13K 10864662 Ki = 80 nM T20401 CY82EF 10865353 Ki = 160 nM T20401 C4E8SG 10865419 Ki = 7 nM T20401 C8M4QY 10865548 Ki = 60 nM T20401 C8OKX5 10865717 Ki = 0.5 nM T20401 C7DV4E 10868086 Ki = 2.9 nM T20401 CQN7G6 10869299 Ki = 33 nM T20401 CP8DF6 10871235 Ki = 286 nM T20401 CUKT63 10872446 Ki = 94 nM T20401 CB3U9M 10874216 Ki = 0.6 nM T20401 C8TM4D 10875038 Ki = 54 nM T20401 C4CM8X 10875810 Ki = 10 nM T20401 CG0Z6I 10876077 Ki = 23 nM T20401 CFXH68 10876514 Ki = 1.1 nM T20401 CT0KQ8 10878827 Ki = 32 nM T20401 C0M3OP 10881177 Ki = 110 nM T20401 CWKM78 10884587 Ki = 24 nM T20401 C23JVY 10886478 Ki = 3 nM T20401 C1YK9S 10886620 Ki = 1.5 nM T20401 C6YGB0 10886642 Ki = 3 nM T20401 CO0V5G 10887065 Ki = 210 nM T20401 C1LX6K 10887220 Ki = 15 nM T20401 CN2L6A 10891750 Ki = 50 nM T20401 CH3LK7 10893334 Ki = 5 nM T20401 CR81KU 10895699 Ki = 12 nM T20401 CY9O1Q 10895884 Ki = 31 nM T20401 CKL08U 10897133 Ki = 61 nM T20401 CBNU79 10897483 Ki = 78 nM T20401 CC51VX 10898100 Ki = 0.6 nM T20401 C9C5HV 10898245 Ki = 0.6 nM T20401 CCW0R7 10899319 Ki = 30.1 nM T20401 C2MY5U 10904482 Ki = 318 nM T20401 CX2K9L 10904983 Ki = 82 nM T20401 C7SH5U 10905170 Ki = 7 nM T20401 CWGB92 10907843 Ki = 23 nM T20401 C2VEZ9 10907925 Ki = 6 nM T20401 C90ZUF 10908674 Ki = 2 nM T20401 CIO06R 10915496 Ki = 78 nM T20401 C0BP2F 10915515 Ki = 38 nM T20401 CG10IV 10916112 Ki = 6 nM T20401 C3WOS1 10917392 Ki = 9800 nM T20401 CUEX85 10918009 Ki = 26 nM T20401 C50OCY 10918511 Ki = 195 nM T20401 C8RXZ0 10919029 Ki = 0.9 nM T20401 C6EPH9 10919571 Ki = 69 nM T20401 CP2Z4G 10919976 Ki = 23 nM T20401 CTDR05 10920174 Ki = 9 nM T20401 C8CV1Z 10923837 Ki = 138 nM T20401 C8TSL7 10926221 Ki = 12 nM T20401 CL5D1P 10926842 Ki = 604000 nM T20401 CVR31W 10930187 Ki = 12 nM T20401 C3WN6P 10931938 Ki = 307 nM T20401 C7FP4E 10932133 Ki = 0.95 nM T20401 CGI4X1 10933094 Ki > 10000 nM T20401 CHZI28 10935067 Ki = 233 nM T20401 C8FIB7 10935528 Ki = 313 nM T20401 CD3GB7 10937101 Ki = 0.8 nM T20401 CO17LZ 10948175 Ki = 52 nM T20401 C8P1ER 10950587 Ki = 66 nM T20401 CZA48D 10952342 Ki = 0.8 nM T20401 CPC86B 10952559 Ki = 145 nM T20401 CZAG71 10952780 Ki = 1 nM T20401 CW2K3M 10953423 Ki = 1600000 nM T20401 CN27BY 10953838 Ki > 100000 nM T20401 C3F9WR 10957702 Ki = 54 nM T20401 CIXO05 10959593 Ki = 0.6 nM T20401 CVG71F 10961747 Ki = 47 nM T20401 CEV7Z1 10962037 Ki = 0.5 nM T20401 CQO1E7 10962986 Ki = 0.9 nM T20401 C5ZPE9 10963315 Ki = 0.6 nM T20401 C0K1QF 10963422 Ki = 31 nM T20401 C4B5DJ 10963712 Ki = 33 nM T20401 C9NC5T 10964817 IC50 = 560000 nM T20401 CCV07P 10970019 Ki = 280 nM T20401 CG08QZ 10970428 Ki = 103 nM T20401 C1H7KL 10970502 Ki = 53 nM T20401 CZPG31 10972292 Ki = 68 nM T20401 C3IDH7 10974944 Ki = 10 nM T20401 CU4TO5 10979790 Ki = 13 nM T20401 CFL46Z 10980153 Ki = 10 nM T20401 C40UVN 10980851 Ki = 81 nM T20401 C59AQM 10983522 Ki = 9 nM T20401 C73HZT 10983658 Ki = 0.3 nM T20401 CM6Z2B 10983679 Ki = 52 nM T20401 C4MXZ2 10985404 Ki = 2 nM T20401 CG61PD 10994426 Ki = 24 nM T20401 CP5A7X 10995068 Ki = 79 nM T20401 CE23PC 10995136 Ki = 0.6 nM T20401 C6VG2U 10995156 Ki = 2 nM T20401 C69NOP 10995214 Ki = 265 nM T20401 COQ4Y6 10995233 Ki = 17 nM T20401 CU91KW 10995327 Ki = 56 nM T20401 C7X4SM 10995402 Ki = 4 nM T20401 C91OEI 10995928 Ki = 13 nM T20401 C8JAX5 10996222 Ki = 215 nM T20401 CIO7M2 10996308 Ki = 9 nM T20401 C60TSD 10996432 Ki = 0.5 nM T20401 CCIT95 11003980 Ki = 0.5 nM T20401 C0R1IV 11004960 Ki = 50 nM T20401 C8YZ0I 11005191 Ki = 57 nM T20401 CVYW37 11006065 Ki = 61 nM T20401 C7WEZ4 11009332 Ki = 62 nM T20401 C1D7XA 11011569 Ki = 54 nM T20401 C9IF1C 11013393 Ki = 125 nM T20401 CEY2A4 11014189 Ki = 88 nM T20401 CD4JQ1 11015176 Ki = 0.7 nM T20401 C2Y6HS 11016006 Ki = 104 nM T20401 CH47PL 11016833 Ki = 2 nM T20401 CNCX57 11017060 Ki = 180 nM T20401 CDR0Y6 11017072 Ki = 1.5 nM T20401 C69TDE 11017073 Ki = 30 nM T20401 C4WU6R 11017835 Ki = 16 nM T20401 C8VI2F 11018004 Ki = 15 nM T20401 C2G5AL 11018133 Ki = 15 nM T20401 CX1F7U 11018241 Ki = 1 nM T20401 C9L3MK 11018318 Ki = 12 nM T20401 CC0F9X 11018319 Ki = 0.5 nM T20401 C6UD9P 11018463 Ki = 8 nM T20401 CAED68 11021701 Ki = 113 nM T20401 CLV4S2 11024707 Ki = 7 nM T20401 CDB16V 11026415 Ki = 0.2 nM T20401 C5CJU7 11028005 Ki = 210 nM T20401 CLM10Q 11028999 Ki = 7 nM T20401 CD8HS3 11031678 Ki = 18 nM T20401 CWO84N 11032771 Ki = 98 nM T20401 CLN35C 11034434 Ki = 45 nM T20401 C36BAC 11034581 Ki > 100000 nM T20401 CFBO12 11035956 Ki = 14 nM T20401 CN6QX1 11036198 Ki = 107 nM T20401 CB4M2O 11036993 Ki = 2 nM T20401 COA8S5 11039158 Ki = 20 nM T20401 CL46GE 11039314 Ki = 0.8 nM T20401 CA1P7Q 11045484 Ki = 80 nM T20401 CV75NH 11047521 Ki = 1 nM T20401 CJ3WY1 11048561 Ki = 280 nM T20401 CVW8K3 11048831 Ki = 310 nM T20401 CC6K7Q 11055293 Ki = 214 nM T20401 COWY75 11055630 Ki = 221 nM T20401 CJ2M4S 11055723 Ki = 125 nM T20401 CO2F4K 11058711 Ki = 70 nM T20401 C3ZP6U 11058734 Ki = 55 nM T20401 CFU60B 11060209 Ki = 3 nM T20401 CC7X2Z 11060668 Ki = 72 nM T20401 CT2D9I 11060771 Ki = 250 nM T20401 C6FA8Y 11060833 Ki = 2 nM T20401 C5X4DW 11060882 Ki = 15 nM T20401 CQBP46 11061197 Ki = 0.89 nM T20401 C1C4OI 11061783 Ki = 7 nM T20401 CP1U3L 11062054 Ki = 10 nM T20401 C36YHJ 11067477 Ki = 235 nM T20401 C8C6ER 11069133 Ki = 0.3 nM T20401 CWM7C8 11071324 Ki = 175 nM T20401 CU5NJ9 11071502 Ki = 310 nM T20401 CRL5I3 11072036 Ki = 19 nM T20401 COGV98 11074431 Ki > 20000 nM T20401 C1BAR9 11077028 Ki = 280 nM T20401 CYT4G0 11078481 Ki = 106 nM T20401 CMQ2Y8 11079355 Ki = 36 nM T20401 CJW7Z3 11081263 Ki = 89 nM T20401 CWTS45 11081678 Ki = 2 nM T20401 CASO94 11081987 Ki = 69 nM T20401 CIC47S 11082122 Ki = 94 nM T20401 C6WU3G 11082240 Ki = 2 nM T20401 C2NXV7 11082357 Ki = 16 nM T20401 CIAW06 11082579 Ki = 0.8 nM T20401 C3O5JB 11083515 Ki = 0.5 nM T20401 C9YZA3 11089252 Ki = 234 nM T20401 CEM9W0 11091166 Ki = 2 nM T20401 CHA42C 11092653 Ki = 110 nM T20401 CS8W3K 11092704 Ki = 200 nM T20401 CSL53A 11093007 Ki = 36 nM T20401 CYST27 11093710 Ki = 10 nM T20401 CMK4Y0 11096006 Ki = 533.6 nM T20401 C2P8ZU 11099090 Ki = 90 nM T20401 CKF5V1 11099458 Ki = 84 nM T20401 C14ZGJ 11101626 Ki = 35 nM T20401 C8DOK1 11102362 Ki = 5 nM T20401 C7RZW3 11103137 Ki = 1.7 nM T20401 COJU46 11103269 Ki = 235 nM T20401 CJF79N 11103375 Ki = 25 nM T20401 CK12PR 11103476 Ki = 13 nM T20401 CWB10K 11103986 Ki = 11.3 nM T20401 C53LWS 11104965 Ki = 13 nM T20401 CZ91PR 11109866 Ki = 97 nM T20401 CYI5F6 11110737 Ki = 210 nM T20401 CVZ89X 11112315 Ki = 227000 nM T20401 CSI1G6 11114605 Ki = 1 nM T20401 CV8S7A 11114620 Ki = 34 nM T20401 C4CE8S 11114939 Ki = 16 nM T20401 CDY1T6 11115104 Ki = 12 nM T20401 CYQ01S 11115351 Ki = 8 nM T20401 CH6IE3 11117198 Ki = 21.5 nM T20401 C9UJ8I 11125027 Ki = 65 nM T20401 C31VGI 11125411 Ki = 1.5 nM T20401 C8X2DC 11127784 Ki = 25.4 nM T20401 C6RM4H 11134231 Ki = 1.5 nM T20401 CU8OF2 11141517 Ki = 300 nM T20401 CZ09RJ 11143896 Ki = 6 nM T20401 CC28PQ 11144024 Ki = 56000 nM T20401 CG36VZ 11144533 Ki = 4 nM T20401 C25CRH 11146161 Ki = 13 nM T20401 CO6X8J 11147037 Ki = 1.5 nM T20401 C5WS3E 11147931 IC50 = 13870 nM T20401 CP3CU4 11157709 Ki = 0.2 nM T20401 CC4IE1 11158128 Ki = 1.21 nM T20401 CPB0A5 11164855 Ki = 5.1 nM T20401 CEYJ94 11165541 Ki = 3.8 nM T20401 C50HJY 11177131 Ki = 13 nM T20401 C3PJ6O 11177505 Ki = 80 nM T20401 CIL4M9 11183499 Ki > 100000 nM T20401 C39IDU 11183936 Ki = 2290 nM T20401 C4W0YX 11186322 Ki = 97 nM T20401 C31DIQ 11188711 Ki = 107 nM T20401 C2CHY5 11188898 Ki = 1470 nM T20401 C5C6MG 11194613 Ki = 570 nM T20401 C5Y1CV 11196316 Ki > 10000 nM T20401 C75FMT 11199252 Ki = 13 nM T20401 CFG37K 11209006 Ki = 0.9 nM T20401 C0P8JA 11215523 Ki = 52 nM T20401 C2AFO0 11216333 Ki = 34 nM T20401 C5L7NR 11217340 Ki = 5900 nM T20401 CJOR84 11220854 Ki = 10 nM T20401 CY2VA5 11221764 Ki = 38 nM T20401 CY1P4Q 11223689 Ki = 7.3 nM T20401 CY9W5K 11226359 Ki = 13 nM T20401 CJQ72W 11230247 IC50 = 71000 nM T20401 C39QJA 11234047 Ki = 1.4 nM T20401 CXAS45 11235150 Ki = 9 nM T20401 C8O1FM 11239393 Ki = 3.74 nM T20401 CHC42Y 11245700 Ki = 14 nM T20401 C92XHG 11245995 Ki = 44 nM T20401 CGE40M 11245996 Ki = 8 nM T20401 CCLV87 11247335 Ki = 18 nM T20401 CN86YV 11250791 Ki = 4.93 nM T20401 CI7YT0 11252120 Ki = 70 nM T20401 C7UVW8 11258440 Ki = 9.8 nM T20401 C12URI 11261582 Ki = 0.39 nM T20401 CIR6A0 11262484 Ki = 4.62 nM T20401 CV7T2K 11269105 Ki = 25 nM T20401 C5P7KN 11269273 Ki = 3.6 nM T20401 C43WCH 11269442 Ki = 15 nM T20401 C7FA3C 11274029 Ki = 4.11 nM T20401 CF1ZC0 11278507 Ki = 9200 nM T20401 CCSA87 11280465 Ki = 30 nM T20401 CF15AS 11287957 Ki = 6775 nM T20401 CG28LP 11290362 Ki = 8300 nM T20401 C0H6GB 11292444 Ki = 12 nM T20401 C1FJ7I 11304583 Ki = 97 nM T20401 C3CDO1 11309586 Ki = 346 nM T20401 CRP08M 11310883 IC50 = 9450 nM T20401 CBC47W 11312414 Ki = 87 nM T20401 CAU4B5 11317320 Ki = 33 nM T20401 CB4U3M 11318985 Ki = 41 nM T20401 CHA0V5 11321514 Ki = 420 nM T20401 CDLR79 11321711 Ki = 15 nM T20401 CA6T0Z 11322287 Ki = 2120 nM T20401 C8ZA1X 11326347 Ki = 12 nM T20401 C84HMR 11329414 Ki = 16 nM T20401 CU73JN 11339017 Ki = 9.5 nM T20401 C8Q5VJ 11342941 Ki = 3.9 nM T20401 CV80KU 11346010 Ki = 5200 nM T20401 CCY4G5 11350445 Ki = 92 nM T20401 CDLS49 11350634 Ki = 61 nM T20401 C3NGH2 11352609 Ki = 19 nM T20401 C8PM3Z 11353795 Ki = 45 nM T20401 C8MI3Z 11361075 Ki = 76 nM T20401 C27RAM 11361542 Ki = 18 nM T20401 CY3B6F 11362509 Ki = 94 nM T20401 CM8Y1J 11367571 IC50 = 8790 nM T20401 CM1XU5 11373291 Ki = 54 nM T20401 C1L2HW 11379214 IC50 = 71000 nM T20401 C6QO0H 11384370 Ki = 9 nM T20401 CY64KU 11385765 Ki = 0.9 nM T20401 CIQ5K7 11387799 Ki = 1.54 nM T20401 C7MK2E 11390955 Ki = 1580 nM T20401 CVT2K6 11396353 Ki = 9.1 nM T20401 CT3E0Y 11399060 Ki = 47 nM T20401 C6RUJ7 11399350 Ki = 1.24 nM T20401 CEO47P 11399506 Ki = 43 nM T20401 CH98MP 11399715 Ki = 1.14 nM T20401 CBVL07 11407223 Ki = 11 nM T20401 C3KV6R 11407281 Ki = 85 nM T20401 C8DF5O 11416806 Ki = 129 nM T20401 CG1A5D 11427826 Ki = 9.6 nM T20401 CGPE75 11428235 Ki = 2.1 nM T20401 CT3NI0 11433608 Ki = 0.21 nM T20401 C3KRG4 11433767 Ki = 3.45 nM T20401 CK7D5V 11438030 Ki = 8400 nM T20401 CUR65I 11441308 Ki = 19 nM T20401 CTU87D 11441601 Ki = 25 nM T20401 C7EOG0 11441729 Ki = 84 nM T20401 C41CHM 11445520 Ki = 27 nM T20401 CMS0Q5 11445529 Ki = 5.96 nM T20401 C32QDC 11453942 Ki = 95 nM T20401 C54AMO 11454377 Ki = 13 nM T20401 C4BQM5 11455128 Ki = 15 nM T20401 C83MCI 11462539 Ki = 20000 nM T20401 C2J9BG 11463026 Ki = 15 nM T20401 CFER43 11467281 Ki = 44 nM T20401 CM9I6W 11467962 Ki = 1.61 nM T20401 CQ1D6E 11470070 IC50 = 9230 nM T20401 CNM06W 11475346 Ki = 15 nM T20401 C91XWJ 11478542 Ki = 52 nM T20401 CIWG06 11479385 Ki = 4.78 nM T20401 CCY54I 11479559 Ki = 4.95 nM T20401 C0WCE4 11482579 Ki = 645000 nM T20401 CL1RC2 11485376 Ki = 1.5 nM T20401 CQ9H8J 11490915 Ki = 40 nM T20401 C4NR1X 11492439 IC50 = 25000 nM T20401 C8QZC4 11499667 IC50 = 48000 nM T20401 C8YO5G 11508929 Ki = 354 nM T20401 CNFY48 11514219 Ki = 10200 nM T20401 CKF6A8 11521331 Ki = 408000 nM T20401 CU8YH7 11533895 Ki = 41 nM T20401 CP8AX2 11540662 Ki = 640 nM T20401 CUT4I6 11550437 IC50 = 21000 nM T20401 CJZ9N8 11573504 Ki = 241 nM T20401 CIMD40 11578176 Ki = 3270 nM T20401 CXB86F 11579563 Ki = 2030 nM T20401 CUJI91 11581618 Ki = 150 nM T20401 CT7LD4 11588141 Ki = 18 nM T20401 CDS25O 11593765 IC50 = 1320 nM T20401 CCB82K 11596108 Ki = 670 nM T20401 CXP21M 11601322 IC50 = 25000 nM T20401 C3FJQ8 11602375 Ki = 230000 nM T20401 CM8P2L 11609292 IC50 = 22 nM T20401 C9QL2F 11615432 Ki = 853.1 nM T20401 C36MZP 11616716 Ki = 6.3 nM T20401 C9JO4B 11623060 IC50 = 30000 nM T20401 CK38DO 11624852 Ki = 18 nM T20401 CV02TF 11632228 Ki = 15 nM T20401 C6MN7Y 11637451 IC50 = 130000 nM T20401 CDU79V 11637531 Ki = 2520 nM T20401 C4EC3U 11663528 Ki = 121 nM T20401 CD1X2V 11666911 IC50 = 100000 nM T20401 C95PYS 11667431 Ki = 1 nM T20401 C9JR2I 11674590 Ki > 100000 nM T20401 CRG49U 11674754 Ki = 7.9 nM T20401 CPGO32 11675510 Ki = 50 nM T20401 C7ZPR9 11681852 Ki = 33 nM T20401 C8F0SQ 11687376 IC50 = 110000 nM T20401 CCG17H 11688636 Ki = 39 nM T20401 CF8IT6 11696964 Ki = 2 nM T20401 CX4W3J 11701693 Ki = 1940 nM T20401 C4VZO5 11709992 Ki = 80 nM T20401 CHAN30 11714982 Ki = 33 nM T20401 C5QIK4 11721174 Ki = 472 nM T20401 C1G0JC 11727638 Ki = 6 nM T20401 CB0EA2 11727760 Ki = 49 nM T20401 CWV01J 11728049 Ki = 80 nM T20401 CJXL89 11728811 Ki = 5 nM T20401 CO03JM 11729079 Ki = 7 nM T20401 CD16NH 11729087 Ki = 69 nM T20401 C0L3RF 11729108 Ki = 7 nM T20401 CV6LK7 11729550 Ki = 36 nM T20401 CYI4S1 11729993 Ki = 26 nM T20401 CH7BF3 11731156 Ki = 43 nM T20401 CE14NA 11731409 Ki = 18 nM T20401 CAW47S 11733056 Ki = 0.6 nM T20401 CEGC64 11735346 Ki = 34 nM T20401 C5YD7H 11735447 Ki = 0.5 nM T20401 CB93NJ 11738933 Ki = 8000 nM T20401 C4FA0T 11740604 Ki = 3 nM T20401 C2D6WI 11748537 Ki = 255 nM T20401 C0TFH3 11760610 Ki = 9 nM T20401 CX5LA8 11763331 Ki = 75 nM T20401 CP78CU 11763512 Ki = 3.13 nM T20401 CBN39F 11767393 Ki = 20 nM T20401 CWM5I6 11773896 Ki = 67 nM T20401 CV68TJ 11774586 Ki = 15 nM T20401 CGUZ16 11776737 IC50 = 6.3 nM T20401 CH7Q5S 11777250 Ki > 10000 nM T20401 C98EGL 11782389 Ki = 844 nM T20401 C9J0YH 11782553 Ki = 50 nM T20401 CJ35OU 11782715 Ki = 53 nM T20401 C37CKB 11782720 Ki = 76 nM T20401 C28PBF 11782912 Ki = 315 nM T20401 CC9L1G 11783323 Ki = 101 nM T20401 C6S8WR 11786209 Ki = 0.3 nM T20401 C4BH9A 11788388 Ki = 883 nM T20401 C7BV5P 11792968 Ki = 11 nM T20401 C4U8QN 11794109 Ki = 6 nM T20401 CW32BE 11794202 Ki = 54 nM T20401 CV7HN1 11795548 Ki = 21 nM T20401 CT2G8Q 11796369 Ki = 9 nM T20401 CG6Z5X 11797062 Ki = 280 nM T20401 C19RCP 11799753 Ki = 100 nM T20401 C07QLV 11800828 Ki = 130 nM T20401 C8X0GK 11800862 Ki = 5 nM T20401 CE1S6W 11801129 Ki = 8 nM T20401 C3E7CX 11801767 Ki = 4 nM T20401 CNB5F6 11802420 Ki = 7 nM T20401 CLC27W 11802422 Ki = 62 nM T20401 C93PTE 11802889 Ki = 15 nM T20401 CH7OA8 11803531 Ki = 2 nM T20401 CSD5K9 11806775 Ki = 138 nM T20401 CL69XF 11809670 Ki = 200 nM T20401 C95JYR 11813616 Ki = 67 nM T20401 C45XIB 11814933 Ki = 13 nM T20401 C0RZ9Y 11816502 Ki = 1.1 nM T20401 C8DY3Z 11817193 IC50 = 7890 nM T20401 C73SVE 11817275 Ki = 75.7 nM T20401 CTR0U7 11823783 Ki = 61 nM T20401 C9CJU1 11824513 Ki = 95 nM T20401 C0VWS3 11824695 Ki = 1.5 nM T20401 CO7K8V 11826660 Ki = 52 nM T20401 C1DB0Z 11828379 Ki = 47 nM T20401 C0OD9Y 11828467 Ki = 71 nM T20401 C18JIA 11828627 Ki = 175 nM T20401 CIWV68 11828670 Ki = 38 nM T20401 CE71FU 11828964 Ki = 0.6 nM T20401 C0CR2G 11848185 Ki = 33 nM T20401 C45NRP 11851425 Ki = 7.6 nM T20401 CJRD82 11966600 Ki = 1 nM T20401 C4T8BS 11967023 Ki = 7 nM T20401 CXSE37 11967046 Ki = 43 nM T20401 C9VM6I 11967472 Ki = 9 nM T20401 CQXG94 11970596 Ki = 310000 nM T20401 CZD0B3 11974341 Ki = 384 nM T20401 C27HSO 11974343 Ki = 44 nM T20401 CCM17V 11974451 Ki = 7.4 nM T20401 CX4IJ0 11974452 Ki = 265 nM T20401 C59UEI 11974453 Ki = 267 nM T20401 CYS7X0 11974454 Ki = 90 nM T20401 C09JGZ 11974455 Ki = 6.8 nM T20401 CS9VL2 11974456 Ki = 218 nM T20401 CP39YI 11974558 Ki = 7 nM T20401 CB97SM 11974559 Ki = 50 nM T20401 CE8WN6 11974560 Ki = 8.1 nM T20401 C06CBY 11974561 Ki = 7.3 nM T20401 CU6K0N 11974562 Ki = 7.3 nM T20401 CI7OE1 11974563 Ki = 470 nM T20401 C6Z5DX 11974630 Ki = 45 nM T20401 CW4X9G 11974631 Ki = 7.5 nM T20401 CEBO65 11974632 Ki = 119 nM T20401 CGQ6B7 11974724 Ki = 423 nM T20401 CHO9T1 11974725 Ki = 8.2 nM T20401 CC8TS1 11974727 Ki = 378 nM T20401 CDL18J 11974728 Ki = 7 nM T20401 C7G3YS 11974830 Ki = 7.2 nM T20401 C1C4JW 11974831 Ki = 8.6 nM T20401 CXW89D 12004261 Ki = 133 nM T20401 C0L4OC 12049163 Ki = 3530 nM T20401 C4ZYQ1 12049713 Ki = 1220000 nM T20401 CNHD71 12051191 Ki > 200000 nM T20401 CMPA32 12066940 Ki > 500000 nM T20401 CB15KR 12066941 Ki > 500000 nM T20401 C2XBZ3 12070806 Ki = 2.4 nM T20401 C32TWU 12094253 Ki = 94.5 nM T20401 CREV05 12140130 Ki = 2270 nM T20401 C6P1VC 12188108 Ki > 10000 nM T20401 C3C9ON 12226066 Ki > 100000 nM T20401 CCY51E 12237458 Ki > 10000 nM T20401 CKI97Z 12344252 IC50 > 200000 nM T20401 C60EFT 12354987 Ki = 120 nM T20401 CPU03D 12355589 Ki = 148 nM T20401 CSYD70 12355590 Ki = 450 nM T20401 C18LXJ 12411101 Ki = 1.9 nM T20401 C0C8FG 12411107 Ki = 95 nM T20401 C5NK2I 12420669 IC50 = 7870 nM T20401 C0JID3 12447203 Ki = 40 nM T20401 CLB1E3 12499681 Ki > 10000 nM T20401 CKSL53 12507616 IC50 > 200000 nM T20401 CP87GR 12516475 Ki = 10.9 nM T20401 C5RS4H 12528487 Ki = 143.8 nM T20401 CM8TP6 12528490 Ki = 1922 nM T20401 C35CMO 12589789 Ki > 10000 nM T20401 CTHQ39 12635073 Ki = 51 nM T20401 CIQX87 12635074 Ki = 19 nM T20401 CK90BP 12765315 Ki = 100100 nM T20401 CZCF65 12914626 Ki = 6000 nM T20401 C1GNM5 12914627 Ki = 750 nM T20401 CO8WC5 12938307 Ki = 4.8 nM T20401 CP70LE 12954894 Ki = 104 nM T20401 COF8W3 13008156 IC50 > 100000 nM T20401 C4IKA3 13087489 Ki > 10000 nM T20401 CF2BM7 13177311 Ki = 7.1 nM T20401 C8VM1A 13201770 Ki = 320 nM T20401 CI31SL 13204988 Ki = 3230 nM T20401 CA2S7W 13236651 IC50 = 3.2 nM T20401 CW3R0Y 13236652 IC50 = 30 nM T20401 CFTU16 13236653 IC50 = 8 nM T20401 CB07AD 13236654 IC50 = 10 nM T20401 CMJ70I 13236655 IC50 = 6 nM T20401 CLIF23 13236656 IC50 = 15 nM T20401 CSD0N8 13236657 IC50 = 6 nM T20401 C6HF1L 13236658 IC50 = 6.8 nM T20401 CPC2I6 13236659 IC50 = 1.6 nM T20401 CZ9W2C 13236661 IC50 = 3.1 nM T20401 C5GAL6 13236662 IC50 = 2 nM T20401 CU67BS 13245460 IC50 = 4 nM T20401 CV1UF4 13306723 Ki = 325 nM T20401 C3ZQW6 13343650 IC50 = 1.8 nM T20401 C85GSD 13360355 Ki = 845 nM T20401 C79BND 13361840 Ki = 678960 nM T20401 CX7M9C 13373975 Ki > 10000 nM T20401 CHC41Q 13381193 Ki > 10000 nM T20401 COLK69 13419352 Ki > 10000 nM T20401 CSN63J 13427336 IC50 = 18180 nM T20401 CX8QE5 13431624 Ki = 48000 nM T20401 CPUJ60 13504187 IC50 = 5.1 nM T20401 CJ37MV 13504188 IC50 = 6.5 nM T20401 CU9Y4F 13504189 IC50 = 6.5 nM T20401 CF5O9P 13504190 IC50 = 3 nM T20401 C8Z3FY 13504191 IC50 = 15 nM T20401 C2HO5Y 13504192 IC50 = 5.5 nM T20401 CR6P1X 13504193 IC50 = 3 nM T20401 C3HOK8 13580495 Ki = 60 nM T20401 CFN29Y 13584466 Ki > 10000 nM T20401 CE5DL6 13617012 IC50 = 5.3 nM T20401 CYI6M2 13617013 IC50 = 6.7 nM T20401 C8L7CZ 13617014 IC50 = 4.6 nM T20401 CQTX49 13738810 IC50 > 10000 nM T20401 C24ABI 13763145 Ki = 3.63 nM T20401 C2JB5Z 13763146 Ki = 28 nM T20401 CC2N6Q 13763149 IC50 = 5 nM T20401 C5FZX9 13763150 IC50 = 100 nM T20401 CR65IU 13763152 Ki = 3.3 nM T20401 C36IXQ 13763155 Ki = 7.11 nM T20401 CZP0T8 13763156 Ki = 1.15 nM T20401 CTHO06 13763157 Ki = 14.2 nM T20401 C4DHA6 13763158 Ki = 30.5 nM T20401 CSY57K 13763159 Ki = 14.1 nM T20401 CC8OY4 13763160 IC50 = 250 nM T20401 C7Q0ZP 13763162 Ki = 18.2 nM T20401 CNP5Z3 13785076 Ki = 1600 nM T20401 C57SFI 13801611 Ki = 647 nM T20401 C24OQJ 13803658 IC50 = 9330 nM T20401 COJ2M1 13911594 IC50 = 3.2 nM T20401 C9L1HM 13911609 Ki = 1.1 nM T20401 CE5MG3 13911613 Ki = 9.3 nM T20401 CBZQ26 13911622 IC50 = 45 nM T20401 C51CST 13911623 Ki = 1.8 nM T20401 C0GQ9U 13911638 Ki = 2.3 nM T20401 CSX0I6 13922809 IC50 = 8.8 nM T20401 COA93E 13922810 IC50 = 12 nM T20401 C4L8SK 13922811 IC50 = 2.6 nM T20401 C5OBY1 13922817 IC50 = 8 nM T20401 C5IOQ7 13922841 IC50 = 23 nM T20401 C3I9ZC 13922842 IC50 = 6.2 nM T20401 CJLM26 13922845 IC50 = 2.6 nM T20401 C06TQG 13922850 IC50 = 18 nM T20401 C5M8PY 13922856 IC50 = 14 nM T20401 C7GC9Y 13922867 IC50 = 9 nM T20401 C3ORS1 13922869 IC50 = 12 nM T20401 CRP48V 13922870 IC50 = 15 nM T20401 C3JUZ0 13922872 IC50 = 10 nM T20401 CVX57O 13922873 IC50 = 9 nM T20401 C45PWL 13922881 IC50 = 6 nM T20401 CY2G9I 13922885 IC50 = 5 nM T20401 CA6YD0 13922891 IC50 = 10 nM T20401 C07HFI 13922894 IC50 = 15 nM T20401 CE6L1Z 13922899 IC50 = 12 nM T20401 C6LT8A 13922900 IC50 = 50 nM T20401 CEGY80 13922901 IC50 = 11 nM T20401 CC25BI 13927398 Ki = 86000 nM T20401 CTYP72 13949092 Ki > 10000 nM T20401 CR6HB5 13949095 Ki > 10000 nM T20401 CFMK94 13949102 Ki > 10000 nM T20401 CL41NJ 13960348 IC50 = 24 nM T20401 CIM6W8 13960351 IC50 = 10000 nM T20401 CVH17I 13960352 IC50 = 700 nM T20401 CAWO49 13960353 IC50 = 20 nM T20401 CN1S7R 13960354 IC50 = 20 nM T20401 C2Q3WJ 13960356 IC50 = 20 nM T20401 C4GO0W 13960357 IC50 = 4.3 nM T20401 CQ9T6Z 13960359 IC50 = 12 nM T20401 C0MDR2 13960360 IC50 = 25 nM T20401 CAB04R 13960362 IC50 = 23 nM T20401 COB6C9 13960369 IC50 = 23 nM T20401 CRI14K 13960370 IC50 = 51 nM T20401 CB6FA5 13960373 IC50 = 900 nM T20401 C9VNA7 13960374 IC50 = 9 nM T20401 C96HGJ 13960375 IC50 = 9 nM T20401 CE2JX7 13960376 IC50 = 3.5 nM T20401 C93SHG 13960377 IC50 = 1.5 nM T20401 C1U0VH 13960378 IC50 = 5 nM T20401 C1PEB8 13960380 IC50 = 4.5 nM T20401 CX5U0D 13960381 IC50 = 4 nM T20401 C7K4JV 14024589 Ki = 1060 nM T20401 C4UG2O 14057643 Ki > 100000 nM T20401 CLS53V 14151811 IC50 = 6160 nM T20401 CQ3D9C 14151815 IC50 > 100000 nM T20401 CNZ6H2 14205726 Ki = 9400000 nM T20401 CTWQ83 14256301 IC50 = 45 nM T20401 C7RUB9 14327005 IC50 = 6 nM T20401 CGJA34 14327007 IC50 = 9 nM T20401 C3R0JV 14327009 IC50 = 11 nM T20401 CIJ6D3 14327011 IC50 = 11 nM T20401 C9BWE3 14327013 IC50 = 11 nM T20401 C1E2TH 14327015 IC50 = 12 nM T20401 C7ZN2H 14327017 IC50 = 8 nM T20401 CNHO79 14327019 IC50 = 14 nM T20401 C4DWC2 14327021 IC50 = 8 nM T20401 C3V0IR 14327023 Ki = 3.4 nM T20401 CK3CP6 14327025 Ki = 8.2 nM T20401 CB56PV 14327027 Ki = 1.24 nM T20401 CT2V9Z 14327029 Ki = 2.6 nM T20401 CCI9S4 14390577 IC50 = 4.8 nM T20401 C3RZ2F 14390578 IC50 = 5.6 nM T20401 C1T0XU 14423973 IC50 = 0.2 nM T20401 CA5Q3H 14425149 Ki = 22171 nM T20401 CXYO59 14435742 IC50 = 8280 nM T20401 C98OYV 14460405 IC50 = 2900 nM T20401 CB59DQ 14460407 IC50 = 2000 nM T20401 CI08OT 14460408 IC50 = 1200 nM T20401 C2JY3N 14460411 IC50 = 480 nM T20401 CJD64R 14460412 IC50 = 400 nM T20401 C1U6AF 14460414 IC50 = 100 nM T20401 C0JO3E 14460415 IC50 = 190 nM T20401 CIY97B 14460418 IC50 = 22 nM T20401 CB8MN4 14460430 IC50 = 12 nM T20401 CCB50P 14460456 IC50 = 2.5 nM T20401 CYU85Z 14460458 IC50 = 10 nM T20401 CSM0B3 14460460 IC50 = 3 nM T20401 CZ3OU4 14460463 IC50 = 3 nM T20401 C6O4FY 14460465 IC50 = 6.3 nM T20401 C8YOU3 14460468 IC50 = 3.3 nM T20401 CAY2P4 14460470 Ki = 3.9 nM T20401 CDIQ70 14460473 IC50 = 4.9 nM T20401 CU1W7A 14460475 IC50 = 6.5 nM T20401 CP32NX 14460477 IC50 = 2.2 nM T20401 CUYQ26 14460478 Ki = 1.92 nM T20401 C0AR8S 14460480 Ki = 1.98 nM T20401 CW0MK2 14460482 Ki = 1.34 nM T20401 CDH0S6 14460484 Ki = 5.5 nM T20401 CH61BI 14460486 Ki = 0.44 nM T20401 C6A2OT 14460488 Ki = 1.1 nM T20401 CS0A7W 14476488 IC50 > 100000 nM T20401 CXS4N1 14476489 IC50 = 16 nM T20401 C3SOX4 14476490 IC50 = 60 nM T20401 C2NT3R 14476491 IC50 = 22 nM T20401 C3S5KB 14476492 IC50 = 30 nM T20401 CJV59W 14476495 IC50 = 25 nM T20401 C92OEB 14498136 Ki = 32.4 nM T20401 CY1GK8 14547488 IC50 = 100 nM T20401 CK4BD7 14601402 Ki = 2.7 nM T20401 COF1W9 14601404 IC50 = 3.2 nM T20401 CNX93C 14601406 IC50 = 2.8 nM T20401 C6NW7Y 14601408 Ki = 0.95 nM T20401 CHOG93 14611919 Ki = 7.2 nM T20401 CR2BE5 14639068 IC50 = 2 nM T20401 CX1BL4 14639069 IC50 = 3.2 nM T20401 C2K4EP 14639075 IC50 = 2.5 nM T20401 CX5S2C 14639076 IC50 = 6.4 nM T20401 CLM37S 14639078 IC50 = 2 nM T20401 CF5EI3 14642289 IC50 = 3.2 nM T20401 CP2J3M 14642290 IC50 = 4.2 nM T20401 CR8A7F 14642291 IC50 = 45 nM T20401 CQ6O2L 14642293 IC50 = 2.5 nM T20401 CQU9G5 14642295 Ki = 6.5 nM T20401 C3FMY4 14642298 IC50 = 5 nM T20401 C5JZ7D 14642299 IC50 = 2.1 nM T20401 C2DT6V 14642300 IC50 = 4.2 nM T20401 CU19HE 14642303 Ki = 2.34 nM T20401 CM1EA0 14700203 IC50 = 8.8 nM T20401 CY1RQ5 14700207 IC50 = 6.6 nM T20401 CD5IK6 14700208 IC50 = 3.2 nM T20401 CY37OF 14700210 Ki = 2.39 nM T20401 C3S7KO 14700211 IC50 = 2.9 nM T20401 CF07XH 14700213 IC50 = 2.9 nM T20401 CZ6SN8 14777102 Ki = 78.7 nM T20401 C76ASY 14787919 Ki > 200000 nM T20401 C35DGV 14873166 Ki > 10000 nM T20401 C9CLH4 14873170 Ki > 10000 nM T20401 C9K0LX 14873174 Ki > 10000 nM T20401 CM34ER 14873177 Ki > 10000 nM T20401 CJZE57 14950175 IC50 = 800 nM T20401 CP0D3K 14950177 IC50 = 1300 nM T20401 CB07FQ 14950178 IC50 = 3 nM T20401 CV0OP3 14950179 IC50 = 200 nM T20401 CW41NT 14950180 IC50 = 2500 nM T20401 CH5YR2 15014351 Ki > 200000 nM T20401 CW3X5A 15038375 Ki = 131000 nM T20401 C7XD2T 15118768 Ki > 100000 nM T20401 CX26PT 15219881 Ki = 12 nM T20401 CK8GE9 15230629 Ki = 2936 nM T20401 C6F3GK 15267134 Ki = 1150.06 nM T20401 CDE4F9 15290967 Ki > 10000 nM T20401 C1IZ7D 15296597 Ki = 120 nM T20401 CJ7V8G 15381187 Ki = 815 nM T20401 C9X6AG 15381192 Ki = 802 nM T20401 CW72MS 15438999 Ki = 36.7 nM T20401 C7R5AH 15476112 Ki = 610 nM T20401 C3CTS0 15523879 Ki = 74.8 nM T20401 CFC2E0 15546406 Ki = 3 nM T20401 C2G4FH 15599374 Ki = 5.5 nM T20401 CQW0U2 15599379 IC50 = 30 nM T20401 C64OPK 15599380 IC50 = 6 nM T20401 C75VGZ 15599382 IC50 = 10 nM T20401 C9P8IS 15599385 IC50 = 5 nM T20401 CP1M9O 15599386 IC50 = 4.5 nM T20401 CT73PL 15618966 Ki = 4.5 nM T20401 CLIO60 15645619 Ki = 2343.9 nM T20401 C80BXE 15669220 Ki = 3.6 nM T20401 CK67AM 15698028 IC50 = 14 nM T20401 CF9Q6I 15698029 IC50 = 4.5 nM T20401 C26QUE 15698030 IC50 = 2.27 nM T20401 COW3F4 15698032 Ki = 2.77 nM T20401 C95JPD 15698040 IC50 = 0.5 nM T20401 C3ANG4 15698041 IC50 = 0.7 nM T20401 C79CSV 15698042 IC50 = 1.15 nM T20401 C36YVX 15707346 IC50 = 9 nM T20401 CZF3L4 15707348 IC50 = 7 nM T20401 CYEJ45 15707349 IC50 = 3 nM T20401 CR1SO6 15707352 IC50 = 18 nM T20401 CYUK73 15707353 IC50 = 6 nM T20401 C6JCN0 15707354 IC50 = 2.3 nM T20401 C5UR2H 15707356 IC50 = 30 nM T20401 CGEO39 15707360 IC50 = 64 nM T20401 C3EM2T 15707361 IC50 = 15 nM T20401 C2QP3F 15707362 IC50 = 8 nM T20401 CAFR14 15707369 IC50 = 20 nM T20401 C8PMQ9 15729847 Ki = 124000 nM T20401 CLT47Z 15783680 Ki > 10000 nM T20401 C6VR7G 15815634 Ki = 86000 nM T20401 C6F0XZ 15818962 Ki > 10000 nM T20401 C8PER5 15938557 Ki > 500000 nM T20401 C3W2MB 15939939 Ki = 6367.7 nM T20401 CB3S7I 16007202 Ki = 87 nM T20401 CM06OZ 16046226 Ki = 19.6 nM T20401 CVZG29 16072592 Ki = 1450 nM T20401 CB73ST 16072595 Ki = 3020 nM T20401 C6U0VS 16078349 Ki = 35 nM T20401 CUT32D 16078350 Ki > 1000 nM T20401 C4JIO0 16078351 Ki = 60 nM T20401 C23FGI 16078837 Ki = 3390 nM T20401 CQ0UX9 16082752 Ki = 94 nM T20401 CBRL45 16082753 Ki = 39 nM T20401 C0BIQ3 16082754 Ki = 61 nM T20401 C6KN4Z 16082755 Ki = 42 nM T20401 C94FZV 16082756 Ki = 64 nM T20401 C85HIK 16082757 Ki = 71 nM T20401 CC74NH 16087011 Ki > 10000 nM T20401 C1CD5B 16087012 Ki > 10000 nM T20401 C8AP5W 16087015 Ki > 10000 nM T20401 CLNI97 16087025 Ki > 10000 nM T20401 CBWD20 16087028 Ki > 10000 nM T20401 CN1XR0 16087029 Ki > 10000 nM T20401 C3GMJ8 16087031 Ki > 10000 nM T20401 CC0Z4V 16119626 Ki > 50000 nM T20401 CB7CU4 16122563 Ki = 23 nM T20401 CV5O8W 16125524 Ki = 8.7 nM T20401 CZ7T4C 16125526 Ki = 46 nM T20401 CS78TE 16125527 Ki = 6.8 nM T20401 C1Z9GQ 16125580 Ki = 7.8 nM T20401 CE4SB2 16125581 Ki = 53 nM T20401 CWM0L9 16125582 Ki = 4.2 nM T20401 C4SD3N 16125583 Ki = 48 nM T20401 CPU0F5 16219477 Ki = 7280 nM T20401 CA6VB3 16221528 Ki = 9400 nM T20401 CQGZ56 16221529 Ki = 10800 nM T20401 C79XIS 16221532 Ki = 10800 nM T20401 CPD68G 16221533 Ki = 11500 nM T20401 CPR94Q 16221534 Ki = 10400 nM T20401 CZO0W5 16221535 Ki = 11400 nM T20401 C0UO9G 16221580 Ki = 9800 nM T20401 CN03IT 16227153 Ki = 78.9 nM T20401 CGB45O 16235229 Ki = 8.9 nM T20401 CV35UO 16450309 IC50 = 36700 nM T20401 CG7OL3 16693908 Ki > 300000000 nM T20401 CMB87O 16717602 Ki > 10000 nM T20401 CC07IS 16718572 IC50 = 97000 nM T20401 COQU32 16729004 Ki = 48 nM T20401 CTK68M 17249579 Ki = 8.9 nM T20401 C5DT7E 17250082 Ki = 162 nM T20401 C6THW2 17268490 Ki = 5005 nM T20401 C5CE8Z 17371280 Ki = 9 nM T20401 CA4OE9 17371576 Ki = 33.8 nM T20401 C73YML 17385730 Ki > 10000 nM T20401 C91LAN 17413757 Ki > 10000 nM T20401 C5M9DR 17433209 Ki > 10000 nM T20401 CYLM41 17492191 Ki > 10000 nM T20401 CDWU20 17537594 Ki = 73.2 nM T20401 CUP95O 17562622 Ki = 0.26 nM T20401 CK7D2I 17748220 Ki = 6 nM T20401 CIR7K0 17751529 IC50 = 17000 nM T20401 CPY2Q0 17751566 IC50 = 130000 nM T20401 C3R0ZH 17751567 IC50 > 1000000 nM T20401 C6EV9N 17751568 IC50 = 85000 nM T20401 CYCI83 17751569 IC50 = 30000 nM T20401 C1MBP4 17751571 IC50 = 29000 nM T20401 CLY1N4 17757567 Ki = 161000 nM T20401 CVN21Y 17770844 Ki = 28880 nM T20401 C3AX8E 17774014 Ki = 49.4 nM T20401 C6SFI8 18268734 Ki = 6.9 nM T20401 CR9VF3 18668331 Ki = 12 nM T20401 CQE5K4 18710120 Ki > 200000 nM T20401 C60NAV 18971452 Ki = 31.7 nM T20401 C6HO7T 18990081 Ki = 184.5 nM T20401 C2K5BX 19374444 Ki = 20.3 nM T20401 CIEH93 19382975 IC50 = 9091 nM T20401 C97MSK 19782950 Ki > 100000 nM T20401 C62PKT 19838794 Ki = 5.7 nM T20401 CU3QS7 19898674 Ki > 10000 nM T20401 CB46JX 20109894 Ki = 1820000 nM T20401 CGE35Q 20182298 Ki = 2.7 nM T20401 CDU40W 20184392 Ki = 60300 nM T20401 CXJ2H4 20195196 Ki = 930 nM T20401 C8Z1CM 20216502 Ki = 58 nM T20401 CAW0I9 20265076 IC50 = 11 nM T20401 C1H6GV 20360268 Ki > 100000 nM T20401 CAG0O1 20368972 Ki = 380 nM T20401 CWX7M9 20426468 IC50 = 2.2 nM T20401 CM8C3U 20426471 IC50 = 10 nM T20401 C8N0DS 20426472 IC50 = 6.8 nM T20401 C15BEG 20694083 Ki = 2200 nM T20401 CKR8T2 20970546 Ki = 4.4 nM T20401 CF28QV 21017876 Ki > 100000 nM T20401 CCJ8Q3 21051266 Ki = 74.3 nM T20401 CH15RE 21051367 Ki = 203 nM T20401 CV34MD 21149346 Ki = 63 nM T20401 CJGU80 21240387 Ki = 97.1 nM T20401 C18KAH 21297028 Ki > 10000 nM T20401 CPG6C1 21416985 Ki = 1070 nM T20401 COG69P 21449436 Ki = 21 nM T20401 C9J1WT 21497848 Ki > 10000 nM T20401 CC5W7X 21542156 Ki > 10000 nM T20401 CD0K1C 21600238 Ki > 10000 nM T20401 C61KUX 21726402 Ki = 88 nM T20401 C54IUM 21778115 Ki = 21470 nM T20401 C27BJH 21778117 Ki = 21160 nM T20401 CJ4O2E 21806575 Ki = 2.7 nM T20401 CO2U7W 21855445 Ki = 81 nM T20401 CZ45AO 21878638 Ki > 10000 nM T20401 C4XAO7 21879009 Ki > 10000 nM T20401 CBS63Q 21879398 Ki > 10000 nM T20401 C02IPY 21978067 Ki = 12.8 nM T20401 C6IZW0 22132896 Ki > 10000 nM T20401 C9U4TE 22313850 Ki = 253 nM T20401 CX4Z1D 22315539 Ki = 136 nM T20401 C81ROV 22316829 Ki = 117 nM T20401 CPR25C 22706805 Ki > 200000 nM T20401 C09ACH 22833027 Ki = 2 nM T20401 C9W4IA 22836851 Ki = 1.8 nM T20401 C4KU1V 22859393 IC50 = 130 nM T20401 CXR35D 22864792 Ki = 5 nM T20401 CWM8S4 22953340 Ki = 3 nM T20401 C2D8ZL 23111570 Ki = 104 nM T20401 CE8C1R 23228497 Ki = 2 nM T20401 C2DOR4 23263451 Ki = 2.4 nM T20401 CYK21X 23274983 IC50 = 5.5 nM T20401 C9KMP4 23275795 Ki = 7.6 nM T20401 CICR37 23426698 Ki = 60170 nM T20401 CY6D4N 23644659 Ki = 9.1 nM T20401 C8UIC6 23644662 Ki = 30 nM T20401 CCLA40 23644663 Ki = 150 nM T20401 CD5KT2 23644664 Ki = 29 nM T20401 C1AVT7 23644700 Ki = 6 nM T20401 C52YRI 23645366 Ki = 9.7 nM T20401 C3BSJ4 23645367 Ki = 8.9 nM T20401 CE50QI 23645368 Ki = 24 nM T20401 CNL51U 23645369 Ki = 9.3 nM T20401 CPRX73 23645370 Ki = 29 nM T20401 CSZ6J4 23645528 Ki = 92 nM T20401 C6UH9Q 23645529 Ki = 38 nM T20401 CD0JP3 23645530 Ki = 45 nM T20401 CM37EC 23645531 Ki = 108 nM T20401 C9PD5F 23645532 Ki > 200 nM T20401 C1OE7R 23645533 Ki = 160 nM T20401 CCSN04 23645534 Ki > 200 nM T20401 CU08WI 23645535 Ki > 200 nM T20401 CY41UC 23645536 Ki > 200 nM T20401 CX15EH 23645537 Ki > 200 nM T20401 CD3Q6G 23645538 Ki > 200 nM T20401 CE6NQ2 23645539 Ki = 15 nM T20401 C4VK3U 23645540 Ki = 9 nM T20401 C8VM1C 23645541 Ki = 190 nM T20401 C0MUT6 23645542 Ki = 9 nM T20401 CNI07H 23645543 Ki = 5 nM T20401 CHK2X1 23645544 Ki = 5 nM T20401 CW1V2Z 23645545 Ki = 4 nM T20401 C6SP7T 23645546 Ki = 44 nM T20401 CD9QO2 23645547 Ki = 0.8 nM T20401 C25YLZ 23645548 Ki = 0.9 nM T20401 C9WT2E 23645682 Ki = 25 nM T20401 CU1OK9 23645683 Ki = 47 nM T20401 CLHE50 23645684 Ki = 124 nM T20401 C0UXY9 23646323 Ki = 279 nM T20401 C3QLX1 23646324 Ki = 128 nM T20401 CMX1A6 23646325 Ki = 7.3 nM T20401 C29HMI 23646326 Ki = 5.8 nM T20401 CA6M4S 23646374 IC50 = 15 nM T20401 CCW81X 23647027 Ki = 9.3 nM T20401 CE20BX 23647028 Ki = 6.9 nM T20401 CNS87E 23661710 Ki = 360000 nM T20401 C8YRU5 23661711 Ki = 2070 nM T20401 CPGY29 23662344 Ki = 8630 nM T20401 C1T3BP 23663627 Ki = 8030 nM T20401 CU3I5E 23664767 Ki = 3220000 nM T20401 CRZT32 23665339 Ki = 30.1 nM T20401 C7V6YP 23665706 Ki > 10000 nM T20401 CH5BD7 23665763 Ki = 89000000 nM T20401 CXWP91 23666732 Ki = 0.95 nM T20401 C6W2BA 23668541 Ki = 73.6 nM T20401 CU08IW 23670409 Ki = 46.7 nM T20401 C1HCX5 23671974 Ki = 51.3 nM T20401 C6F9NR 23672331 Ki = 93000 nM T20401 C21XEP 23672490 Ki = 320000 nM T20401 CYO7C3 23673162 Ki = 113000 nM T20401 CZNV20 23673832 Ki = 100000 nM T20401 CDB01O 23674157 Ki > 2000 nM T20401 C4UFA0 23674499 Ki = 350000 nM T20401 CPI26E 23677888 Ki = 1960 nM T20401 CR7O3Q 23677931 Ki = 4 nM T20401 CKL59B 23679442 Ki = 45.1 nM T20401 CNIF07 23681162 Ki = 7280 nM T20401 CJA07G 23685506 Ki = 6790 nM T20401 CC93FA 23686905 Ki = 0.7 nM T20401 CZD6O0 23688497 Ki = 293 nM T20401 C54XWY 23689557 Ki = 4360 nM T20401 CH0QD2 23690451 Ki = 3340 nM T20401 C45EHX 23690537 Ki = 83000 nM T20401 C7LE5M 23690998 Ki = 4700 nM T20401 CE52UX 23691027 Ki = 3810 nM T20401 CE91KL 23691977 Ki = 298 nM T20401 CBU67Z 23691979 Ki = 5850 nM T20401 CE03MX 23692005 Ki = 110000 nM T20401 CK2Q0I 23697126 Ki = 107 nM T20401 C4XE6Y 23699059 Ki = 3330 nM T20401 C7U8GK 23699988 IC50 = 6.8 nM T20401 CR41LS 23703293 Ki = 103000 nM T20401 CPX0I4 24204718 Ki = 421 nM T20401 CF83JT 24204719 Ki = 276 nM T20401 CSWR58 24204720 Ki = 297 nM T20401 CIQ9L6 24204924 Ki = 408 nM T20401 CL2V5T 24204925 Ki = 419 nM T20401 C14RLU 24204932 Ki = 275 nM T20401 CN5ST6 24206002 Ki = 415 nM T20401 CPD4Z6 24206003 Ki = 510 nM T20401 C1Y2JB 24286289 Ki = 89.2 nM T20401 CKE1A3 24416843 Ki = 19.4 nM T20401 CBXC05 24424330 IC50 = 29 nM T20401 CA3Y8I 24588559 Ki = 234 nM T20401 CG98KI 24588612 Ki = 258 nM T20401 CK79DN 24588735 Ki = 173 nM T20401 CGHW54 24640576 Ki = 43.2 nM T20401 C01LHS 24640776 Ki = 3.8 nM T20401 CT8O2Z 24643222 Ki = 2 nM T20401 CB6WE3 24650532 Ki = 2.5 nM T20401 C1I9HZ 24692821 Ki = 28.1 nM T20401 CQG9O0 24816432 Ki = 10 nM T20401 CX10RQ 24823136 Ki = 235 nM T20401 CAS51H 24823137 Ki = 13 nM T20401 CXV0A1 24823299 Ki = 2.1 nM T20401 CK0D4U 24823300 Ki = 380 nM T20401 CU6VO3 24823301 Ki = 460 nM T20401 C8A9PE 24823302 Ki = 7.5 nM T20401 C5W7AC 24823303 Ki = 9.1 nM T20401 CZMT56 24823304 Ki = 8.7 nM T20401 CB9U5Z 24823476 Ki = 440 nM T20401 CXT1C5 24823477 Ki = 427 nM T20401 CBDO71 24823478 Ki = 8.2 nM T20401 CUT3V8 24823479 Ki = 6.7 nM T20401 C3UYV0 24823480 Ki = 432 nM T20401 CJQ3M4 24823631 Ki = 13 nM T20401 CPQN52 24823632 Ki = 7.6 nM T20401 CN75LK 24823633 Ki = 2.3 nM T20401 C8D1GQ 24829374 Ki = 300000 nM T20401 CV5YR0 24843241 Ki = 1.2 nM T20401 C4C1LK 24853952 Ki > 300000 nM T20401 C4OJ8T 24853953 Ki = 300000 nM T20401 CX3E5U 24853954 Ki > 300000 nM T20401 CNR3U7 24866945 IC50 > 10000 nM T20401 CQRZ10 24877657 Ki = 18 nM T20401 CCOG78 24944524 Ki = 51940 nM T20401 C15OJW 24966977 Ki = 730 nM T20401 CQ9B0P 24970303 IC50 = 31 nM T20401 C2JQ7M 25040103 Ki = 549 nM T20401 C62DIS 25048179 Ki = 802 nM T20401 CTVO94 25071013 Ki = 7.7 nM T20401 CB0E2M 25071014 Ki = 8.4 nM T20401 COI25U 25131351 Ki = 18 nM T20401 CNMY17 25131685 Ki = 198 nM T20401 CP67CK 25134300 IC50 = 31 nM T20401 CGW49I 25146686 IC50 > 40000 nM T20401 CB7V8Y 25147773 Ki = 4.2 nM T20401 CG0S7T 25154732 Ki = 540 nM T20401 CYG1H9 25154741 Ki = 820 nM T20401 CZ3EI0 25174192 IC50 = 47 nM T20401 C3KF1V 25178145 Ki = 65 nM T20401 C8PMK7 25178356 Ki = 63 nM T20401 C9HZG2 25181078 Ki = 8.4 nM T20401 CMYP34 25181079 Ki = 9.3 nM T20401 C7U1YC 25181080 Ki = 57 nM T20401 C85HLG 25181081 Ki = 35 nM T20401 C4M9XV 25242508 Ki = 12100 nM T20401 CU14KG 25258358 Ki > 200000 nM T20401 CQ1WE2 25258360 Ki > 200000 nM T20401 CL5EZ6 25258361 Ki = 41100 nM T20401 COU19V 25258363 Ki > 200000 nM T20401 C5T1NZ 25294048 Ki = 50.5 nM T20401 CRP6F5 25335375 Ki = 6.3 nM T20401 CPN2T5 25392418 Ki = 7.1 nM T20401 C1AOB3 25981084 Ki = 0.83 nM T20401 CP02LF 26365005 Ki = 3.8 nM T20401 C0RF4D 26470767 Ki > 100000 nM T20401 CMUT78 26500397 Ki = 5.1 nM T20401 C5EC2T 26535209 Ki = 3 nM T20401 CLNR46 26598995 Ki = 2337 nM T20401 CA9UZ7 26773685 Ki = 0.79 nM T20401 C39JBI 27868037 Ki = 2.6 nM T20401 C8KQ5N 27868059 Ki = 85 nM T20401 CQSA29 27868075 Ki = 1765 nM T20401 C7QB8M 27868953 Ki = 26.2 nM T20401 CWU2R0 27869227 Ki = 1.9 nM T20401 C46OQT 27869236 Ki = 6.5 nM T20401 C85HLF 27869237 Ki = 31.4 nM T20401 C5OWP7 27869350 Ki = 3725 nM T20401 CF02EA 27869546 Ki = 22.7 nM T20401 C1G3XO 27869982 Ki = 1290 nM T20401 C8ML3W 27870055 Ki = 2634 nM T20401 C5RX6E 27870091 Ki = 2.7 nM T20401 CMK25I 27870443 Ki = 226 nM T20401 CQK4O6 27870796 Ki = 1060 nM T20401 C2Z4FP 27870803 Ki = 75 nM T20401 C7ZT8O 27871218 Ki = 0.3 nM T20401 C61AIY 28452155 Ki = 701.8 nM T20401 C3RG8K 28846439 Ki = 24.2 nM T20401 C4EB0J 29034199 Ki = 2.6 nM T20401 C0CJ5I 29045530 Ki = 86.6 nM T20401 CF8SA7 29559803 Ki = 2.3 nM T20401 C4R0ZU 29981063 Ki > 10000 nM T20401 CBPO08 34751720 Ki = 704.3 nM T20401 CVXO26 35053285 Ki = 10 nM T20401 CF3HA1 35871284 Ki = 34.1 nM T20401 CI0K1J 36865965 Ki = 5.7 nM T20401 C5IUO9 38154971 Ki = 17.2 nM T20401 CZE95V 38155699 Ki = 24.9 nM T20401 CSB4C7 38159448 Ki = 258 nM T20401 C4F7YT 40086402 Ki > 10000 nM T20401 C06EUO 40662472 Ki = 14.6 nM T20401 C1U4TL 41180562 Ki = 9 nM T20401 CH2P6W 41430216 Ki = 2485 nM T20401 C5YBO2 41484755 Ki = 908 nM T20401 CUK13R 41874556 Ki > 10000 nM T20401 C0J8DM 42597612 Ki = 4350 nM T20401 C8A5CF 42597613 Ki = 4550 nM T20401 C58ZUN 42597614 Ki = 3920 nM T20401 COG2A0 42597615 Ki = 4510 nM T20401 C1J9CQ 42597616 Ki = 3900 nM T20401 COG2I5 42598921 Ki = 4980 nM T20401 CDXS12 42598922 Ki = 4100 nM T20401 C6WU8M 42609905 Ki = 17 nM T20401 CP7UM8 42643988 Ki = 276000 nM T20401 C0IE3B 42644449 Ki = 618000 nM T20401 CT2C3D 42644450 Ki = 382000 nM T20401 CYJ0H4 43089860 Ki = 6.1 nM T20401 CNB1E8 43139163 Ki = 142.5 nM T20401 CXJY80 43235186 Ki = 0.63 nM T20401 CC5TY6 43321518 Ki = 5329 nM T20401 C23CNV 43321585 Ki = 141.5 nM T20401 C7EO2A 43329592 Ki = 27.8 nM T20401 CA0DX4 43342474 Ki = 23.8 nM T20401 C2HY4R 43342475 Ki = 7.8 nM T20401 CBK0M6 43342481 Ki = 1.4 nM T20401 C41VHR 43468983 Ki = 15.7 nM T20401 C82MRL 44144383 Ki = 72.5 nM T20401 CUT9E0 44186130 Ki = 8 nM T20401 C8D7UR 44186132 Ki = 6 nM T20401 CL08CN 44186134 Ki = 6.7 nM T20401 C3UC8S 44186136 Ki = 6.6 nM T20401 CXT6O8 44186138 Ki = 1.01 nM T20401 CLP2V8 44186201 Ki = 0.96 nM T20401 CEN2Y5 44186203 Ki = 7.8 nM T20401 CYR23T 44186205 Ki = 1.8 nM T20401 CAF52T 44186207 Ki = 0.88 nM T20401 CZR5W4 44186209 Ki = 6.9 nM T20401 C4POV2 44186263 Ki = 6.5 nM T20401 CW95CB 44186265 Ki = 0.96 nM T20401 CQ6JB5 44186267 Ki = 0.97 nM T20401 C1REF8 44186269 Ki = 6.8 nM T20401 CZM6N5 44186271 Ki = 3.6 nM T20401 CMR52W 44201382 IC50 = 26.6 nM T20401 CIG89O 44201383 IC50 = 48 nM T20401 CCXN08 44219644 IC50 = 15 nM T20401 C82GHC 44219651 Ki = 330 nM T20401 CW1Q9E 44219652 IC50 = 250 nM T20401 C49UTC 44219653 IC50 = 130 nM T20401 C36OBU 44219661 IC50 = 100 nM T20401 CI2LS6 44221745 Ki = 7.6 nM T20401 CAY8B9 44221746 Ki = 57 nM T20401 CP1K7W 44221747 Ki > 100000 nM T20401 CFEJ21 44221748 Ki > 100000 nM T20401 CZ9X2W 44221749 Ki = 51 nM T20401 C8T4IC 44221941 Ki = 8025 nM T20401 CJE2D7 44221942 Ki = 7.2 nM T20401 CERA26 44221943 Ki = 4.9 nM T20401 C7TJF2 44221944 Ki > 100000 nM T20401 CVJ5A1 44246262 Ki = 105 nM T20401 CZKG76 44246264 Ki = 104 nM T20401 C3E0CZ 44246268 Ki = 105 nM T20401 C0QZI4 44246269 Ki = 107 nM T20401 CZL01D 44246271 Ki = 109 nM T20401 CN6T0X 44266037 Ki = 0.3 nM T20401 C8U6RP 44266090 Ki = 0.17 nM T20401 CGO28Y 44266117 Ki = 1 nM T20401 CG2D4X 44268930 Ki = 2 nM T20401 CX1CK5 44268931 Ki = 6 nM T20401 CZT39W 44268932 Ki = 48 nM T20401 C6ECO2 44268933 Ki = 33 nM T20401 C15VUL 44268934 Ki = 6 nM T20401 CO83EW 44269005 Ki = 0.5 nM T20401 C8T3FR 44269010 Ki = 1.4 nM T20401 C9LUN8 44269014 Ki = 780 nM T20401 C5HTZ4 44269015 Ki = 13 nM T20401 CE07DX 44269023 Ki = 6 nM T20401 CD71PZ 44269025 Ki = 40 nM T20401 CM1SO2 44269027 Ki = 11 nM T20401 CIZ2H8 44269028 Ki = 150 nM T20401 C53OWA 44269034 Ki = 790 nM T20401 C0Y8PD 44269040 Ki = 7 nM T20401 CJ4CQ2 44269056 Ki = 15 nM T20401 CHQT54 44269066 Ki = 48 nM T20401 CARG97 44269072 Ki = 18 nM T20401 CB59ZH 44269073 Ki = 55 nM T20401 CZ5G4I 44295070 Ki = 450 nM T20401 CZH4J1 44295071 Ki = 450 nM T20401 C4TKI3 44295073 Ki = 5 nM T20401 C5N9HB 44295232 Ki = 36 nM T20401 C5SJ8L 44295325 Ki = 85 nM T20401 C8V4GI 44295335 Ki = 330 nM T20401 C63FNX 44295336 Ki = 420 nM T20401 CFQ3Z0 44295339 Ki = 73 nM T20401 CNR6G2 44295340 Ki = 79 nM T20401 CM1V4E 44295349 Ki = 400 nM T20401 C9G5AI 44295381 Ki = 53 nM T20401 C7R6JT 44295382 Ki = 36 nM T20401 CWFN72 44295388 Ki = 11 nM T20401 C1K8SN 44295397 Ki = 21 nM T20401 CM7AJ8 44295411 Ki = 51 nM T20401 CYBT62 44295448 Ki = 44 nM T20401 C20PFZ 44295453 Ki = 50 nM T20401 C13NTV 44295458 Ki = 85 nM T20401 CUIB83 44295459 Ki = 240 nM T20401 C0AGJ6 44295464 Ki = 38 nM T20401 C2N6AL 44295477 Ki = 250 nM T20401 C1RVC6 44295493 Ki = 250 nM T20401 CGAJ68 44295497 Ki = 210 nM T20401 CF8Q3E 44295519 Ki = 10 nM T20401 C38CMP 44295539 Ki = 16 nM T20401 C9K8WR 44295565 Ki = 305 nM T20401 CE49OS 44295574 Ki = 490 nM T20401 CV1LQ8 44295581 Ki = 73 nM T20401 CEV72P 44295589 Ki = 300 nM T20401 C7C5BP 44295596 Ki = 520 nM T20401 C18IXK 44295597 Ki = 290 nM T20401 C6WG1X 44295602 Ki = 410 nM T20401 CU4O3K 44295612 Ki = 62 nM T20401 C6J3EG 44295620 Ki = 120 nM T20401 CAQ28E 44295627 Ki = 280 nM T20401 C90FBC 44295647 Ki = 305 nM T20401 CB2J7Q 44295734 Ki = 7 nM T20401 C8B1EU 44295749 Ki = 9 nM T20401 CAQ8D5 44295756 Ki = 3 nM T20401 C5Z7KR 44295772 Ki = 12 nM T20401 C8SE3Z 44295795 Ki = 45 nM T20401 CCI7X0 44295824 Ki = 340 nM T20401 C8MVP1 44295825 Ki = 275 nM T20401 C4M1WH 44295835 Ki = 9 nM T20401 CYM91I 44295843 Ki = 43 nM T20401 CJ0S8N 44295871 Ki = 75 nM T20401 CH36RU 44295906 Ki = 74 nM T20401 CWY05P 44295942 Ki = 110 nM T20401 CFZN67 44295943 Ki = 115 nM T20401 CC68PJ 44295959 Ki = 66 nM T20401 CG14BN 44295994 Ki = 74 nM T20401 CGCE21 44296010 Ki = 72 nM T20401 C1VKH3 44296089 Ki = 52 nM T20401 COGP36 44296104 Ki = 40 nM T20401 C68EID 44296814 Ki = 1.49 nM T20401 C64EZD 44296918 Ki = 3.4 nM T20401 C6V9WT 44309709 Ki = 15 nM T20401 CYUE74 44309710 Ki = 27 nM T20401 CERI42 44309802 Ki = 1.6 nM T20401 CLBU37 44310092 Ki = 29 nM T20401 CW0S8U 44311169 Ki = 15 nM T20401 C0B4HZ 44312333 Ki > 200 nM T20401 C76HLZ 44314854 Ki = 1.37 nM T20401 C91HDR 44315566 Ki > 10000 nM T20401 C4T7BJ 44322528 Ki = 3 nM T20401 CV72ZF 44322583 Ki = 15 nM T20401 CG0RI3 44322584 Ki = 20 nM T20401 CXDA80 44322970 Ki = 2 nM T20401 CLQS83 44327323 Ki = 0.3 nM T20401 CPTU85 44329131 Ki = 3.1 nM T20401 C7X5HT 44329132 Ki = 4 nM T20401 CK2O4V 44329147 Ki = 1.9 nM T20401 CEU58D 44329411 Ki = 1.3 nM T20401 CNLO86 44329422 Ki = 4.6 nM T20401 CI6AW0 44329423 Ki = 1.7 nM T20401 C6DKW1 44329437 Ki = 2 nM T20401 C3RFO4 44329445 Ki = 1.7 nM T20401 CI9KS2 44329453 Ki = 2.8 nM T20401 CU78BY 44329463 Ki = 1.8 nM T20401 CX2HZ1 44329466 Ki = 2.4 nM T20401 CR13HU 44329471 Ki = 2.9 nM T20401 C7U0QG 44329472 Ki = 1.7 nM T20401 COZ8Q4 44329485 Ki = 5.1 nM T20401 CC85EH 44329560 Ki = 1.4 nM T20401 CNY0R6 44329561 Ki = 1.5 nM T20401 CX0W5V 44329576 Ki = 5.9 nM T20401 C6BGE3 44329679 Ki = 2 nM T20401 CP67GZ 44329699 Ki = 1.6 nM T20401 CM21EZ 44329700 Ki = 2.1 nM T20401 CQY2H4 44329734 Ki = 2.9 nM T20401 CPG0U9 44329736 Ki = 3.1 nM T20401 C4D9HU 44329737 Ki = 5.4 nM T20401 CU41NJ 44329768 Ki = 3.3 nM T20401 CS7D6E 44329771 Ki = 5.2 nM T20401 CBK4M3 44329804 Ki = 2.2 nM T20401 C7G4IN 44329805 Ki = 2.9 nM T20401 CH43UT 44332605 Ki = 4 nM T20401 CWRD02 44332665 Ki = 3 nM T20401 CP0WO3 44338600 Ki = 1.5 nM T20401 C3A0RM 44345919 Ki = 20 nM T20401 CFJD87 44345920 Ki = 900 nM T20401 CU3Y7S 44345997 Ki = 0.44 nM T20401 CW08NK 44345998 Ki = 1.1 nM T20401 CV5PG7 44345999 Ki = 1.58 nM T20401 C3XJK5 44346012 Ki = 1200 nM T20401 CX1IL7 44346124 IC50 = 1.2 nM T20401 CVRZ98 44346142 IC50 = 3.2 nM T20401 C32GKC 44346246 IC50 = 3 nM T20401 CKI8S2 44347455 Ki = 64 nM T20401 C3T5BJ 44347553 Ki = 5 nM T20401 CK62UO 44347554 Ki = 8 nM T20401 CFHX13 44347728 Ki = 73 nM T20401 C8MJ2U 44347729 Ki = 8 nM T20401 CKA91T 44347760 Ki = 68 nM T20401 CCJ82U 44347774 Ki = 61 nM T20401 C0ZAW1 44347825 Ki = 1.3 nM T20401 C4O3KI 44347826 Ki = 40 nM T20401 CUT7R6 44347834 Ki = 41 nM T20401 C18YIR 44347836 Ki = 3 nM T20401 CL53AZ 44347837 Ki = 3 nM T20401 C0AXH3 44347849 Ki = 3 nM T20401 CLXC41 44347889 Ki = 50 nM T20401 CR0X1H 44347896 Ki = 3 nM T20401 C3WA6I 44347907 Ki = 9 nM T20401 CRU7E6 44347909 Ki = 4 nM T20401 C0VS9L 44347924 Ki = 57 nM T20401 CNAV57 44359667 Ki = 3571083.46 nM T20401 CWO45K 44359689 Ki = 32232945.95 nM T20401 C01LBE 44359718 Ki = 111173172.7 nM T20401 CY8LR9 44359736 Ki = 35710834.58 nM T20401 C01RDP 44359753 Ki = 7575302.85 nM T20401 C39VNB 44359757 Ki = 111173172.7 nM T20401 CB52DJ 44359768 Ki = 100000000 nM T20401 C30JRF 44359802 Ki = 23812226.23 nM T20401 CS52CH 44359804 Ki = 83329734.86 nM T20401 CJS09K 44359815 Ki = 30304002.98 nM T20401 C2EY0I 44359830 Ki = 66665324.9 nM T20401 C4T6SW 44359832 Ki = 0.3 nM T20401 CH95PU 44359930 Ki = 100000000 nM T20401 CS09NE 44359982 Ki = 4000368.51 nM T20401 CL6WK9 44359987 Ki = 2 nM T20401 C3WSX6 44360017 Ki = 22724796.35 nM T20401 CXBM69 44360292 Ki = 3 nM T20401 CQ3G7E 44363244 Ki = 5 nM T20401 C83HZB 44363263 Ki = 4 nM T20401 C5NGZ6 44363316 Ki = 15 nM T20401 C6T7KR 44363320 Ki = 25 nM T20401 CXG27B 44363365 Ki = 3 nM T20401 CL8QM1 44363386 Ki = 12 nM T20401 C8GC9V 44363414 Ki = 12 nM T20401 CB2JK5 44363440 Ki = 5 nM T20401 C6ETL2 44363444 Ki = 5 nM T20401 CT8QU4 44363445 Ki = 7 nM T20401 C0DTE3 44363462 Ki = 15 nM T20401 CITL93 44363515 Ki = 8.913 nM T20401 C5I2YQ 44363519 Ki = 10 nM T20401 CH4YN1 44363520 Ki = 6 nM T20401 CM6O2J 44363524 Ki = 3 nM T20401 C9S6NA 44363540 Ki = 3.981 nM T20401 COQM57 44363589 Ki = 5 nM T20401 C10PKB 44363655 Ki = 4 nM T20401 CL8OU3 44363657 Ki = 3 nM T20401 CYE04Z 44363692 Ki = 1 nM T20401 C1IM4R 44363714 Ki = 8 nM T20401 CA40KV 44363764 Ki = 3.981 nM T20401 CDN4K1 44363803 Ki = 5 nM T20401 CAPN36 44367390 Ki = 4500 nM T20401 CS4P3F 44367405 Ki = 2.7 nM T20401 CD98KU 44367410 Ki = 23 nM T20401 CF8J7B 44367431 Ki = 13 nM T20401 CE18VJ 44367432 Ki > 10000 nM T20401 CT0R9B 44367463 Ki = 4.7 nM T20401 CHE0B6 44373668 Ki = 275 nM T20401 CLQK83 44373669 Ki = 30 nM T20401 CZ01KF 44373682 Ki = 250 nM T20401 CLA0S6 44373694 Ki = 145 nM T20401 CY9NC0 44373699 Ki = 33 nM T20401 C1NT8P 44373700 Ki = 45 nM T20401 C8LSM2 44373716 Ki = 8 nM T20401 CGRJ30 44373728 Ki = 36 nM T20401 C0T5BN 44373729 Ki = 6 nM T20401 CJ4HY3 44373738 Ki = 3 nM T20401 CCQ89X 44373741 Ki = 0.5 nM T20401 CI34UE 44373906 Ki = 270 nM T20401 C4B7LG 44373919 Ki = 125 nM T20401 C63UGJ 44373942 Ki = 120 nM T20401 CPG1U2 44373981 Ki = 8 nM T20401 C3SQF9 44373982 Ki = 12 nM T20401 CH8F9D 44373983 Ki = 18 nM T20401 CU9O5K 44377610 IC50 = 25 nM T20401 CKM68G 44377611 IC50 = 9 nM T20401 CFD32U 44377632 IC50 = 210 nM T20401 CX3Z6C 44377760 IC50 = 11 nM T20401 CDE9A8 44377914 IC50 = 110 nM T20401 COZ45V 44377929 IC50 = 32 nM T20401 CIX89D 44380403 Ki > 100000 nM T20401 CR8UH5 44380428 Ki = 21000 nM T20401 CZHX52 44380431 Ki = 71 nM T20401 CJVY96 44380588 Ki = 17 nM T20401 CCLG64 44380603 Ki = 27 nM T20401 CBC73O 44380656 Ki = 15000 nM T20401 C4M7PV 44380677 Ki > 100000 nM T20401 CT3CM0 44380678 Ki = 25000 nM T20401 CM0V9I 44380939 Ki = 36 nM T20401 CXY9F6 44380940 Ki = 49 nM T20401 C3XN9Y 44380951 Ki = 21 nM T20401 CUV2W6 44380955 Ki = 19 nM T20401 CKT4J7 44381089 Ki = 68 nM T20401 C1M4GF 44381090 Ki = 13000 nM T20401 C6K9PD 44381123 Ki > 100000 nM T20401 CVB7U8 44381140 Ki = 890 nM T20401 C5O9LH 44389667 Ki = 18 nM T20401 CL5GF2 44389703 Ki = 6 nM T20401 C9DRN1 44389734 Ki = 14 nM T20401 CE9BS6 44389758 Ki = 9 nM T20401 C68TCP 44389772 Ki = 10 nM T20401 C9OM5F 44389791 Ki = 13 nM T20401 C7VMQ6 44389836 Ki = 75 nM T20401 CF19RI 44389844 Ki = 150 nM T20401 CG2U5A 44389881 Ki = 13 nM T20401 CR16DV 44389954 Ki = 27 nM T20401 C8KE4X 44389960 Ki = 7 nM T20401 CEV89Z 44389961 Ki = 7 nM T20401 C5ZCF3 44389968 Ki = 48 nM T20401 C06AUB 44389978 Ki = 8 nM T20401 C09EFT 44389990 Ki = 6 nM T20401 CFBU06 44389993 Ki = 19 nM T20401 C3IBQ1 44389995 Ki = 16 nM T20401 CP8JK3 44390019 Ki = 12 nM T20401 CWCQ49 44390027 Ki = 159 nM T20401 CVW6E1 44390031 Ki = 11 nM T20401 C5TO9D 44390032 Ki = 185 nM T20401 CI8PB1 44391626 Ki = 6 nM T20401 C68BRH 44391633 Ki = 15 nM T20401 C6BUC8 44391791 Ki = 77 nM T20401 CWR3F1 44391802 Ki = 165 nM T20401 CM6F7X 44391805 Ki = 3.8 nM T20401 C93OPV 44391820 Ki = 1.8 nM T20401 CDH40E 44391824 Ki = 1.6 nM T20401 CUK9X4 44391833 Ki = 1.9 nM T20401 COTH27 44391859 Ki = 265 nM T20401 CD9H6W 44392389 Ki = 15 nM T20401 C5ZA9R 44395106 Ki = 27 nM T20401 C4OR5F 44395107 Ki = 36 nM T20401 C9J2ME 44395133 Ki = 21 nM T20401 C9MLB4 44395134 Ki = 278 nM T20401 CI3O9B 44395149 Ki = 23 nM T20401 CO8J7I 44395150 Ki = 15 nM T20401 CPB8W7 44395163 Ki = 13 nM T20401 C8EK1N 44395173 Ki = 130 nM T20401 CQ54DL 44395174 Ki = 98 nM T20401 CWUP51 44395202 Ki = 20 nM T20401 CIWO28 44395243 Ki = 112 nM T20401 CYR62U 44395244 Ki = 21 nM T20401 CUW0D8 44395258 Ki = 23 nM T20401 C6H1QR 44395691 Ki = 0.6 nM T20401 CWN75T 44395718 Ki = 0.6 nM T20401 CR81IG 44395747 Ki = 0.5 nM T20401 CYS09N 44395778 Ki = 1.7 nM T20401 CMSJ40 44395790 Ki = 12 nM T20401 CD4AX9 44395811 Ki = 3.4 nM T20401 CX9RC2 44395866 Ki = 0.7 nM T20401 CN7A1U 44395892 Ki = 0.8 nM T20401 C90XMR 44395897 Ki = 0.9 nM T20401 CVC7K9 44395919 Ki = 0.9 nM T20401 CL5FR8 44396970 Ki = 11 nM T20401 CY4L9G 44396983 Ki = 20 nM T20401 C3CB6J 44397074 Ki = 5 nM T20401 CWBC15 44397108 Ki = 16 nM T20401 C3VG4H 44397112 Ki = 46 nM T20401 C65XZL 44397209 Ki = 5 nM T20401 CFK1W2 44397213 Ki = 5 nM T20401 CX1V2T 44397238 Ki = 7 nM T20401 C6Y5MJ 44397294 Ki = 8 nM T20401 C5Z7FC 44397318 Ki = 4 nM T20401 CA65VH 44398374 Ki = 50 nM T20401 C7T8XG 44399285 Ki = 46 nM T20401 CNSR28 44399286 Ki = 77 nM T20401 C8NOW9 44399298 Ki = 14 nM T20401 C89LNG 44399317 Ki = 18 nM T20401 CT3V7P 44399318 Ki = 450 nM T20401 CCD34Q 44399321 Ki = 35 nM T20401 C67HFO 44399335 Ki = 49 nM T20401 CQJZ93 44399338 Ki = 5.5 nM T20401 C0KFU7 44399339 Ki = 6.3 nM T20401 CH6GT7 44399340 Ki = 5.1 nM T20401 CG0Z9A 44399346 Ki = 175 nM T20401 C8EQG2 44399347 Ki = 83 nM T20401 C5GJ3N 44399351 Ki = 33 nM T20401 CNTM52 44399371 Ki = 38 nM T20401 C3QZR6 44399393 Ki = 62 nM T20401 C7BHR6 44399404 Ki = 31 nM T20401 C7LCX4 44399427 Ki = 33 nM T20401 C48MQR 44399437 Ki = 146 nM T20401 CCZG27 44399440 Ki = 21 nM T20401 C72HQK 44399449 Ki = 9.8 nM T20401 CGEX61 44399456 Ki = 124 nM T20401 CU1B9T 44399459 Ki = 216 nM T20401 CV9EU2 44399460 Ki = 326 nM T20401 CQCB53 44399461 Ki = 338 nM T20401 CZ4DF9 44399462 Ki = 32 nM T20401 CZ3YC5 44399486 Ki = 23 nM T20401 CVK1X8 44399489 Ki = 50 nM T20401 CUK37Q 44399499 Ki = 65 nM T20401 CVP43X 44399501 Ki = 39 nM T20401 CRM73I 44399515 Ki = 27 nM T20401 CK6G2Y 44399516 Ki = 596 nM T20401 C4UEG1 44399517 Ki = 765 nM T20401 CL6F3X 44399532 Ki = 83 nM T20401 CU7BK9 44399535 Ki = 28 nM T20401 CX6B8J 44399541 Ki = 63 nM T20401 CMFY95 44399542 Ki = 36 nM T20401 C8B9NK 44399547 Ki = 138 nM T20401 CT57KL 44399549 Ki = 16 nM T20401 CB0R2P 44399570 Ki = 163 nM T20401 CD5MJ6 44399571 Ki = 29 nM T20401 C3EBD7 44399585 Ki = 5.1 nM T20401 C0RT3E 44399598 Ki = 5.4 nM T20401 CPKG57 44399624 Ki = 3.1 nM T20401 CI5Y0H 44399639 Ki = 5 nM T20401 C2T7MB 44399654 Ki = 48 nM T20401 CU3DY1 44399655 Ki = 32 nM T20401 C4AD1R 44399664 Ki = 5.2 nM T20401 CR95YM 44399687 Ki = 5.1 nM T20401 CGC2M5 44399695 Ki = 5.1 nM T20401 C3W9CF 44399734 Ki = 5.1 nM T20401 CUXT35 44401673 Ki = 12 nM T20401 C4AD6B 44401689 Ki = 180 nM T20401 C1A5NV 44401728 Ki = 10.3 nM T20401 CWJ08B 44401743 Ki = 8300 nM T20401 C9O1UL 44401744 Ki = 313 nM T20401 C27YCF 44401745 Ki = 50.5 nM T20401 C83EIL 44401769 Ki = 290 nM T20401 C2HDZ6 44401810 Ki = 9900 nM T20401 CJ86PU 44401826 Ki = 8.1 nM T20401 C0F1VY 44401832 Ki = 9100 nM T20401 CQ02ZD 44401833 Ki = 8200 nM T20401 C5PR9E 44401857 Ki = 220 nM T20401 C7NM9T 44401871 Ki = 9100 nM T20401 CD9I8V 44401873 Ki = 89.6 nM T20401 CYQF42 44401889 Ki = 7.2 nM T20401 CIN38J 44401926 Ki = 301000 nM T20401 C75WFG 44401951 Ki = 230000 nM T20401 CX1LH3 44401952 Ki = 278 nM T20401 CIO61G 44401975 Ki = 129000 nM T20401 C9M0ID 44401978 Ki = 7900 nM T20401 CU53CI 44401994 Ki = 473 nM T20401 C34PLI 44402062 Ki = 251000 nM T20401 CF6X9Y 44402148 Ki = 10.1 nM T20401 C28JBO 44402274 Ki = 290 nM T20401 CGPF38 44402275 Ki = 46 nM T20401 CT6UF5 44402709 Ki = 14 nM T20401 C5FC0Y 44402716 Ki > 1000 nM T20401 C8N0GW 44402748 Ki = 55 nM T20401 C9AJ7Z 44402772 Ki = 21 nM T20401 CR72VG 44402825 Ki = 102 nM T20401 C5LU4G 44403258 Ki = 8.3 nM T20401 C6OS3R 44403265 Ki = 6 nM T20401 CI18FK 44403266 Ki = 436 nM T20401 CR2Z7F 44403267 Ki = 475 nM T20401 C0W6BQ 44403268 Ki > 1000 nM T20401 C8QXA6 44403278 Ki > 1000 nM T20401 CSN79Y 44403312 Ki = 82 nM T20401 CW93DL 44405187 Ki = 32 nM T20401 CSXF07 44405190 Ki = 104 nM T20401 CQN4P8 44408881 Ki = 104 nM T20401 COM50H 44408887 Ki = 94 nM T20401 CVJ5T9 44416166 Ki = 19.9 nM T20401 CZT1U9 44416167 Ki = 5570 nM T20401 CQ36IP 44416168 Ki = 18.5 nM T20401 CS49FE 44416185 Ki = 547 nM T20401 CEH5P1 44416186 Ki = 806 nM T20401 C8C4IJ 44416203 Ki > 10000 nM T20401 CE6N7Q 44416215 Ki > 10000 nM T20401 CY9VT1 44416239 Ki = 8.6 nM T20401 CI01QM 44416240 Ki = 3800 nM T20401 CX8ZQ9 44416241 Ki = 2675 nM T20401 CRX27F 44416256 Ki > 10000 nM T20401 C68YLB 44416306 Ki = 244 nM T20401 C5ROE2 44416307 Ki = 9.2 nM T20401 C47OTU 44416317 Ki = 536 nM T20401 CE4M9P 44416378 Ki = 4620 nM T20401 CE03DL 44416379 Ki = 6100 nM T20401 C67IEM 44420782 Ki = 7.6 nM T20401 CY49HT 44423674 Ki = 8700 nM T20401 CHI5G1 44423675 Ki = 96 nM T20401 CFC3M6 44423676 Ki = 4200 nM T20401 CO24JF 44423677 Ki = 91 nM T20401 C7F9DB 44423678 Ki = 97 nM T20401 CJ6GW5 44423679 Ki = 96 nM T20401 CUKM29 44423680 Ki = 95 nM T20401 C3R0FS 44423681 Ki = 94 nM T20401 C14DBJ 44423682 Ki = 9600 nM T20401 CA90GQ 44424362 Ki > 200000 nM T20401 C5HB4P 44424363 Ki > 200000 nM T20401 CK8S7Y 44424364 Ki > 200000 nM T20401 C28QYE 44424366 Ki > 200000 nM T20401 CP3OY8 44428369 Ki = 12.5 nM T20401 CM3J0U 44430517 Ki = 10 nM T20401 C9LT7Y 44430518 Ki = 62 nM T20401 C1VTB6 44430520 Ki = 750 nM T20401 C2L5MB 44430521 Ki = 11 nM T20401 CVEO17 44430523 Ki = 8 nM T20401 C8MFL1 44430524 Ki = 9 nM T20401 CW8DJ9 44435841 Ki = 9200 nM T20401 CQ4RC2 44435843 Ki = 354000 nM T20401 C9RYT1 44435845 Ki = 2670 nM T20401 CHDA78 44435846 Ki = 350000 nM T20401 C1G7HL 44435848 Ki = 412000 nM T20401 CW3M0X 44435849 Ki = 13460 nM T20401 CA4ZH8 44435850 Ki = 235750 nM T20401 CW73VG 44435851 Ki = 3830 nM T20401 C3D6AL 44435853 Ki = 433000 nM T20401 C6X5NI 44435855 Ki = 2150 nM T20401 COUY42 44435856 Ki = 9250 nM T20401 C1LM4Y 44435857 Ki = 3690 nM T20401 CU72AI 44435858 Ki = 3680 nM T20401 C5AMH4 44435861 Ki = 346000 nM T20401 C38GXC 44435862 Ki = 3890 nM T20401 C1AOX2 44435863 Ki = 11250 nM T20401 CFBT23 44435864 Ki = 3540 nM T20401 C37DRO 44435865 Ki = 2830 nM T20401 CT3S5B 44435866 Ki = 13250 nM T20401 C3PTQ7 44435867 Ki = 8850 nM T20401 CUO81X 44445087 Ki = 10 nM T20401 CE61WS 44445088 Ki = 5 nM T20401 COS30Z 44445089 Ki = 110 nM T20401 CWGV59 44445090 Ki = 100 nM T20401 CGP58E 44445091 Ki = 20 nM T20401 C72RWK 44445092 Ki = 10 nM T20401 CV4WU5 44445094 Ki = 15 nM T20401 C74ECN 44448778 Ki = 42 nM T20401 CX50NI 44448882 Ki = 41 nM T20401 CNRW48 44448977 Ki = 33 nM T20401 CUWK18 44449006 Ki = 20 nM T20401 CB9KU0 44449032 Ki = 47 nM T20401 CSFE58 44449055 Ki = 152 nM T20401 CV31AN 44449057 Ki = 12 nM T20401 C7PU2N 44449080 Ki = 37 nM T20401 CLIV87 44449082 Ki = 28 nM T20401 C48XSU 44449083 Ki = 165 nM T20401 C53DYE 44458870 Ki = 17 nM T20401 C7ULS2 44459273 Ki = 2 nM T20401 C23QZG 44459307 Ki = 1.5 nM T20401 C8P4EB 44459430 Ki = 149 nM T20401 CNW10Y 44459431 Ki = 3.8 nM T20401 CM24YZ 44461366 IC50 = 2 nM T20401 CR6BU2 44461673 IC50 = 1.2 nM T20401 CSYX03 44461779 IC50 = 2.8 nM T20401 CNEQ96 44461795 IC50 = 4 nM T20401 C5TQG4 44461813 IC50 = 1.2 nM T20401 CC8X4S 44461814 IC50 = 1.2 nM T20401 C9ABT5 44461815 IC50 = 3.5 nM T20401 C7TCS9 44461827 IC50 = 1.4 nM T20401 CJI1P9 44461839 IC50 = 32 nM T20401 C54IPC 44461840 IC50 = 25 nM T20401 CGY35K 44461906 IC50 = 2.9 nM T20401 C9V3RL 44461907 IC50 = 3.2 nM T20401 CG6J7D 44461913 IC50 = 2.1 nM T20401 C7ZPH3 44461922 IC50 = 4.1 nM T20401 COAZ80 44461923 IC50 = 1.8 nM T20401 C71MCO 44461927 IC50 = 4 nM T20401 C4AOE5 44461957 IC50 = 1.6 nM T20401 CU7KE6 44462114 IC50 = 4 nM T20401 CF5E8J 44462115 IC50 = 60 nM T20401 C1TVZ8 44469864 IC50 = 1300 nM T20401 C1NTS9 44470705 Ki = 14000 nM T20401 CUER27 44511333 IC50 = 65100 nM T20401 CFW8V2 44520897 Ki = 390 nM T20401 CR4NZ3 44520898 Ki = 50 nM T20401 CI78UO 44520899 Ki = 52 nM T20401 CQUC34 44520900 Ki = 51 nM T20401 CNC1D8 44520905 Ki = 97 nM T20401 CR43NP 44520906 Ki = 51 nM T20401 C92QWL 44521066 IC50 = 86 nM T20401 CHCT21 44542292 Ki = 4.7 nM T20401 CG61YX 44542293 Ki = 38.2 nM T20401 CL8AQ5 44542294 Ki = 10.5 nM T20401 CF2RX4 44542600 Ki = 8.6 nM T20401 C5MZ3O 44542742 Ki = 4.2 nM T20401 CI9VZ6 44542743 Ki = 49.3 nM T20401 C8E0MV 44552472 Ki = 813 nM T20401 CKG53H 44552473 Ki = 447 nM T20401 C17XAJ 44552559 Ki = 561 nM T20401 C18XNW 44564181 Ki = 2610 nM T20401 CQIJ49 44564248 Ki = 265 nM T20401 CR8V7Q 44564282 Ki = 380 nM T20401 CJ05ZA 44571847 Ki = 1080 nM T20401 C52WIF 44571892 Ki = 940 nM T20401 C64APD 44574189 Ki = 15700 nM T20401 CV5XS1 44574190 Ki = 10710 nM T20401 CE0ZS5 44574217 Ki = 5300 nM T20401 C3OYU7 44574218 Ki = 4240 nM T20401 CHJV65 44574219 Ki = 14980 nM T20401 C4FI0H 44574220 Ki = 10770 nM T20401 CM9E2T 44574221 Ki = 3820 nM T20401 C5MCT7 44574248 Ki = 600 nM T20401 CZB19D 44574249 Ki = 9310 nM T20401 C48VUR 44574250 Ki = 11300 nM T20401 CL96KM 44574828 Ki = 1560 nM T20401 C0AD8M 44574829 IC50 = 55 nM T20401 CGQ1I9 44574914 IC50 = 10 nM T20401 CH03WX 44577410 Ki = 470 nM T20401 CCH53K 44577411 Ki = 378 nM T20401 CACY16 44577574 Ki = 10.7 nM T20401 CQ3RT6 44577575 Ki = 11.7 nM T20401 C03CLH 44577576 Ki = 8.3 nM T20401 CKT85S 44577800 Ki = 7.9 nM T20401 C3DU8S 44577801 Ki = 18.6 nM T20401 CZ29UX 44577802 Ki = 33.8 nM T20401 C5RZK3 44577803 Ki = 8.1 nM T20401 CB1E6X 44577804 Ki = 40.3 nM T20401 CCW3S1 44578981 Ki = 79 nM T20401 CU7Y8T 44578982 Ki = 12 nM T20401 C86YLD 44579460 Ki = 16 nM T20401 CD4WO8 44579535 Ki = 36 nM T20401 CF0KQ8 44581932 Ki = 2 nM T20401 CXD9V3 44590306 Ki = 55700 nM T20401 CM2L4W 44591861 Ki = 7.8 nM T20401 CSU20V 44591862 Ki = 8.7 nM T20401 CF9MS6 44591908 Ki = 8.7 nM T20401 CQ40FB 44592373 Ki = 5.3 nM T20401 C15THP 44592446 Ki = 5.4 nM T20401 CDB3X7 44592447 Ki = 6.9 nM T20401 C2J3ER 44592448 Ki = 9.9 nM T20401 CUXJ39 44592449 Ki = 6.8 nM T20401 CTI2C1 44592450 Ki = 5.3 nM T20401 COS6N0 44592512 Ki = 5.6 nM T20401 CASL51 44592513 Ki = 7.8 nM T20401 CXL68J 44592514 Ki = 7.6 nM T20401 COL03N 44592515 Ki = 6.2 nM T20401 CHMW14 44592516 Ki = 2.9 nM T20401 CS9M6N 44597633 IC50 = 300000 nM T20401 CQOF25 44597634 IC50 = 45000 nM T20401 CWG4S1 44629933 Ki = 49200000 nM T20401 CVB2U3 44632018 Ki = 15 nM T20401 COX6D8 45028566 Ki = 90 nM T20401 CF2WL9 45028890 Ki = 95 nM T20401 C4MO3S 45028891 Ki = 56 nM T20401 C80CDA 45028892 Ki = 98.3 nM T20401 C6YHW4 45028893 Ki = 50.5 nM T20401 C16ILW 45028894 Ki = 97 nM T20401 C5W1RK 45029305 IC50 = 7590 nM T20401 C6T3IO 45029333 IC50 = 6440 nM T20401 CEY71Z 45117541 Ki = 1280 nM T20401 C0JD8L 45260265 IC50 = 8.4 nM T20401 C64AJS 45261768 IC50 = 22 nM T20401 C2WMZ9 45261770 IC50 = 9 nM T20401 CP3L0D 45261775 IC50 = 9 nM T20401 C9LC8Y 45261786 IC50 = 9 nM T20401 CF6MR9 45261797 IC50 = 16 nM T20401 COB68P 45261808 IC50 = 14 nM T20401 CF65OV 45261822 IC50 = 11 nM T20401 C2Z7TP 45261834 IC50 = 8 nM T20401 C1N7XY 45261845 IC50 = 26 nM T20401 C8ES6W 45261846 IC50 = 4.8 nM T20401 CMCL90 45264429 IC50 = 2.5 nM T20401 CZV1M4 45265042 IC50 = 9 nM T20401 C9JMG4 45265045 IC50 = 15 nM T20401 CN14ZE 45265147 IC50 = 2.4 nM T20401 COF3J5 45265148 IC50 = 12 nM T20401 CHI19Y 45265159 IC50 = 36 nM T20401 C59KZS 45265160 IC50 = 12 nM T20401 C7M2GB 45265187 IC50 = 29 nM T20401 CJ93XZ 45265192 IC50 = 23 nM T20401 C7L3DB 45265194 IC50 = 5 nM T20401 C0RA9D 45265200 IC50 = 4.5 nM T20401 CPQ30H 45265216 IC50 = 4 nM T20401 CUQB41 45266944 IC50 = 243000 nM T20401 C2SHJ7 45266999 Ki > 100000 nM T20401 COE8U0 45267045 Ki > 10000 nM T20401 CM20PR 45267196 Ki = 27600 nM T20401 CA07CZ 45268031 Ki = 438 nM T20401 C3VB9U 45268767 IC50 = 790000 nM T20401 C23MVW 45269009 IC50 = 59 nM T20401 C0RG8K 45269749 Ki = 8800 nM T20401 CPF1T6 45272409 IC50 = 331 nM T20401 CJX37G 45375967 Ki = 14 nM T20401 CJ68EO 45375968 Ki = 13 nM T20401 CSE48D 45375973 Ki = 63 nM T20401 C4LZW6 45483195 Ki = 32.4 nM T20401 C2K1GS 45483207 Ki = 24 nM T20401 C6E7XJ 45484068 Ki = 4500 nM T20401 CGI25L 45484069 Ki = 4350 nM T20401 CVG6K1 45484072 Ki = 4910 nM T20401 CV5RQ3 45484187 Ki = 59 nM T20401 CTG20B 45485271 Ki = 72300 nM T20401 CK4U0V 45485283 Ki = 22700 nM T20401 CW7FR9 45486144 Ki = 71 nM T20401 C8T4WM 45486167 Ki = 76 nM T20401 C5GZ1B 46197458 Ki = 14.8 nM T20401 C3Z7OL 46197569 Ki = 13.4 nM T20401 CUQF42 46197571 Ki = 15.5 nM T20401 C4C7XG 46197572 Ki = 13.1 nM T20401 CLBG91 46197677 Ki = 14.8 nM T20401 C9GC5Q 46197678 Ki = 16.3 nM T20401 C16XCV 46197680 Ki = 58.8 nM T20401 C3JW1R 46197790 Ki = 62.5 nM T20401 CD49XQ 46197791 Ki = 9.1 nM T20401 C4H9TD 46197792 Ki = 7.8 nM T20401 C0W1GZ 46197794 Ki = 5 nM T20401 CUO20Q 46197893 Ki = 4.8 nM T20401 CN7KI3 46197894 Ki = 14.5 nM T20401 CD74LO 46197895 Ki = 13.3 nM T20401 CZ93SW 46197897 Ki = 12 nM T20401 CNQZ73 46197997 Ki = 15.1 nM T20401 CCAX25 46197998 Ki = 15.4 nM T20401 CQ3R2U 46197999 Ki = 73.8 nM T20401 CGM42H 46198111 Ki = 56.2 nM T20401 C0DKY8 46198112 Ki = 15.2 nM T20401 CBWN61 46198113 Ki = 7.8 nM T20401 C0AF1L 46198114 Ki = 7.6 nM T20401 C1KWB5 46198220 Ki = 4.6 nM T20401 CEV26X 46198221 Ki = 5.2 nM T20401 C1ALN3 46201612 Ki = 8640 nM T20401 CHE08Y 46225608 Ki = 2310 nM T20401 CIE2H3 46225609 Ki = 2440 nM T20401 CF42NR 46225631 Ki = 496 nM T20401 C0ZG3L 46225639 Ki = 524 nM T20401 CGW1I5 46225644 Ki = 472 nM T20401 CEOQ06 46225645 Ki = 648 nM T20401 CR0WO3 46225646 Ki = 734 nM T20401 CC2BL5 46225656 Ki = 785 nM T20401 CW52PZ 46225672 Ki = 343 nM T20401 CXJ1C9 46225673 Ki = 536 nM T20401 C6ION5 46236927 Ki = 9.6 nM T20401 C7SFG3 46236928 Ki = 237 nM T20401 CC82QE 46237039 Ki = 258 nM T20401 CBCK34 46237040 Ki = 321 nM T20401 CSD29O 46237041 Ki = 190 nM T20401 CEB1X9 46237042 Ki = 142 nM T20401 C1VIK9 46237043 Ki = 106 nM T20401 C3RJ5M 46237044 Ki = 233 nM T20401 CU5Y9E 46237045 Ki = 10.1 nM T20401 CM7N6J 46237172 Ki = 104 nM T20401 CP15GJ 46237173 Ki = 10.3 nM T20401 C25FBC 46567082 Ki = 17.9 nM T20401 CQN8K4 46635132 Ki = 42.1 nM T20401 CA4FJ2 46703925 Ki = 45.8 nM T20401 C2WB4C 46703927 Ki = 94.8 nM T20401 CO2IU4 46704079 Ki = 52 nM T20401 CB85EQ 46704080 Ki = 88.3 nM T20401 CAE9Z3 46704081 Ki = 46.1 nM T20401 CD5V6T 46704082 Ki = 117 nM T20401 CQ0YA8 46830113 Ki = 12 nM T20401 CEJ2L7 46830114 Ki = 25 nM T20401 C5MB8F 46845029 IC50 = 73100 nM T20401 C8MR0H 46847340 IC50 = 100 nM T20401 CRS8J6 46860267 Ki = 3310 nM T20401 C2RA7G 46861342 Ki = 3.6 nM T20401 CCW34G 46861804 IC50 = 45.9 nM T20401 CRZ29M 46861805 IC50 = 3.77 nM T20401 CI21XG 46861806 IC50 = 8.29 nM T20401 C2S4YC 46866644 IC50 = 820 nM T20401 C7QR8Y 46866645 IC50 = 580 nM T20401 CUH07J 46866646 IC50 = 100 nM T20401 C8GK4C 46866647 IC50 = 310 nM T20401 CT65RE 46868356 Ki > 10000 nM T20401 C7CQ6I 46871755 Ki = 13 nM T20401 CNEO10 46871889 Ki = 3640 nM T20401 C7UKN2 46884029 Ki = 18.1 nM T20401 C1DCM9 46884093 Ki = 65.8 nM T20401 C4ALG9 46884132 Ki = 7.1 nM T20401 CTRY21 46884169 Ki = 16.2 nM T20401 CBM20W 46884215 Ki = 62.7 nM T20401 CR61DW 46884254 Ki = 4.7 nM T20401 CH14SG 46884922 Ki = 10 nM T20401 CFK1L8 46884953 Ki = 18 nM T20401 C9QVN3 46884954 Ki = 14 nM T20401 CT9OQ6 46887904 IC50 = 12.3 nM T20401 CVX05D 46887935 IC50 = 21.3 nM T20401 CZ23PM 46887936 IC50 = 35.9 nM T20401 C6QT5B 46887937 IC50 = 10.1 nM T20401 CTL5J9 46887938 IC50 = 106 nM T20401 CNT04P 46887939 IC50 = 84.1 nM T20401 C6EZM9 46887969 IC50 = 67.6 nM T20401 CTM4O2 46887970 IC50 = 20.2 nM T20401 CCGD62 46887971 IC50 = 21.5 nM T20401 CBMK80 46887972 IC50 = 16.5 nM T20401 C2Z0FD 46887973 IC50 > 5000 nM T20401 C1BW9J 46887974 IC50 = 20 nM T20401 C9KMN4 46888010 IC50 = 2710 nM T20401 C52NDI 46888011 IC50 = 57.1 nM T20401 C5H0YK 46888012 IC50 = 26.7 nM T20401 CP0O7K 46888057 IC50 = 23.2 nM T20401 C6TXO0 46888058 IC50 = 19.9 nM T20401 CVU6W4 46888059 IC50 = 2.19 nM T20401 C53URE 46888060 IC50 = 25.8 nM T20401 CIC14R 46888061 IC50 = 10.6 nM T20401 CS0J9F 46888093 IC50 = 34.6 nM T20401 C51JUC 46888094 IC50 = 18.4 nM T20401 C7W2QG 46888095 IC50 = 11.5 nM T20401 CV49AY 46888096 IC50 = 79.3 nM T20401 CEAQ12 46888136 IC50 = 52.8 nM T20401 CLT61J 46888137 IC50 = 321 nM T20401 CFLG09 46888138 IC50 = 386 nM T20401 C5I0CN 46888139 IC50 = 2.79 nM T20401 C60IQZ 46888469 IC50 = 110000 nM T20401 CD4LT3 46888470 IC50 = 98100 nM T20401 CW94IO 46888471 IC50 = 113000 nM T20401 CE19LY 46888472 IC50 = 86300 nM T20401 C2X6AE 46888473 IC50 = 129000 nM T20401 CZY28W 46888518 Ki = 15135612.48 nM T20401 C0AN1G 46890958 Ki = 31 nM T20401 C08WJF 46890959 Ki = 28 nM T20401 C9UK8S 46891017 Ki = 25 nM T20401 C2KT4I 46891018 Ki = 47000 nM T20401 C93AIR 46899573 Ki = 112000 nM T20401 C4GZ6A 46907387 Ki = 56.9 nM T20401 CJ0R2O 46911381 Ki = 8 nM T20401 C6YK2E 46913624 Ki = 920 nM T20401 CAF1K0 46913625 Ki = 37100 nM T20401 CO60NB 46918149 Ki = 350 nM T20401 C9T3WF 46933594 Ki = 172 nM T20401 C1WE2D 46933744 Ki = 112 nM T20401 CUHI56 46933745 Ki = 108 nM T20401 C27DFQ 46933746 Ki = 114 nM T20401 CSQG87 46933747 Ki = 106 nM T20401 C08BKN 46933748 Ki = 105 nM T20401 C54PRX 46933749 Ki = 103 nM T20401 CP62AV 46933896 Ki = 102 nM T20401 C03FQY 46943413 Ki = 66.1 nM T20401 C31ZQL 49843495 Ki = 55 nM T20401 CQJX35 49843496 Ki = 16 nM T20401 CQA97T 49844531 Ki = 70 nM T20401 CN2U1Z 49844532 IC50 = 80 nM T20401 C5SWC2 49844677 Ki = 190 nM T20401 CD73OF 49844678 IC50 = 260 nM T20401 C56KLI 49844679 IC50 = 590 nM T20401 CR87DE 49844829 Ki = 50 nM T20401 CCOB94 49929067 Ki = 3.5 nM T20401 CY45IU 49957432 IC50 = 2.09 nM T20401 C5Z2QA 50741845 Ki = 774 nM T20401 CVC35K 50899076 IC50 = 8600 nM T20401 CR3I2H 50899077 IC50 = 9660 nM T20401 CEHP41 50909907 Ki = 15 nM T20401 CB4O0Y 50909908 Ki = 3.3 nM T20401 CU9S2J 50939824 Ki = 707 nM T20401 CCM82N 50939825 Ki = 480 nM T20401 C1QBZ3 50942416 Ki = 2.1 nM T20401 C62ZDQ 51035422 Ki = 37 nM T20401 CW0CJ2 51035423 Ki = 41 nM T20401 C5CR2F 51039206 Ki = 11.3 nM T20401 C3SH7R 51039207 Ki = 11.3 nM T20401 C4MWO1 51039208 Ki = 11.3 nM T20401 CS5ZR3 51039209 Ki = 11.3 nM T20401 C8TR3Z 51047320 Ki = 3.4 nM T20401 CHK5G9 51059586 Ki > 50000 nM T20401 CDP03R 51076628 Ki = 0.3838 nM T20401 C5BA0P 51346838 Ki = 1773 nM T20401 C8G3WE 51346839 Ki = 398 nM T20401 CQUS34 51347355 IC50 = 5000 nM T20401 C8XGV5 51349458 Ki = 11.3 nM T20401 C4S5NC 51349459 Ki = 11.3 nM T20401 CZH4T2 51349599 Ki = 11.3 nM T20401 CK3U6Q 51349600 Ki = 11.3 nM T20401 CDF2V8 51349601 Ki = 754 nM T20401 CC2OT0 51349602 Ki = 11.3 nM T20401 CSOX94 51349603 Ki = 11.3 nM T20401 CG26DK 51349604 Ki = 513 nM T20401 CUP39M 51355749 Ki = 9600 nM T20401 CJ1M5T 51355750 Ki = 64.7 nM T20401 CBL9U1 51356010 Ki = 9.7 nM T20401 CLG43P 51669707 IC50 = 8280 nM T20401 C1FM4S 52940811 Ki = 553 nM T20401 CE15GD 52941031 Ki = 286 nM T20401 CE7WD6 52942084 Ki = 475 nM T20401 CRMY05 52942168 Ki = 620 nM T20401 C7OA0E 52942246 Ki = 574 nM T20401 C4O3HF 52942279 Ki = 260 nM T20401 C2OQL5 52942476 Ki > 100000 nM T20401 C0R5HD 52943223 Ki = 538 nM T20401 CCNT92 52943270 Ki = 243 nM T20401 CXMY91 52943276 Ki = 70 nM T20401 CC67HN 52943455 Ki = 516 nM T20401 C50ELG 52943614 Ki > 100000 nM T20401 C7HU5Q 52944525 Ki = 10 nM T20401 CB4UY1 52944603 Ki = 391 nM T20401 C3G6WM 52944864 Ki > 100000 nM T20401 C20FAL 52945268 Ki = 352 nM T20401 C3MLZ1 52945326 Ki = 518 nM T20401 CBGN39 52945721 Ki = 256 nM T20401 CCV6U5 52945740 Ki = 247 nM T20401 CX28EM 52945837 Ki = 45 nM T20401 C6ZCQ2 52947045 Ki = 9 nM T20401 CRVI93 52948047 Ki > 100000 nM T20401 CDNI78 52948211 Ki = 10 nM T20401 CAW78K 52948213 Ki = 196 nM T20401 CA59GT 52948974 Ki = 205 nM T20401 C14WUN 52949402 Ki = 604 nM T20401 CW92IL 52949544 Ki = 127 nM T20401 CLK0S1 52950139 Ki = 26400 nM T20401 CPGW70 53245686 Ki = 28 nM T20401 CF89ML 53307609 Ki = 35450 nM T20401 C60FVH 53317618 Ki = 2459 nM T20401 C7FJN3 53318913 Ki = 1563 nM T20401 CPSU85 53320228 Ki = 2254 nM T20401 C6VN4G 53320229 Ki = 2304 nM T20401 CKRO12 53321135 Ki = 104 nM T20401 CTF92V 53322463 Ki = 82 nM T20401 CQ8R0Y 53322880 Ki = 1207 nM T20401 CA80RT 53322881 Ki = 1165 nM T20401 CTMG14 53322882 Ki = 78.9 nM T20401 C8Z2IL 53324362 Ki = 93 nM T20401 C9PDY6 53326762 Ki = 963 nM T20401 CK4ZG3 53342705 Ki = 1.896 nM T20401 CHF62Q 53361485 IC50 = 1410 nM T20401 CJ3F4R 53361486 IC50 = 2660 nM T20401 C08REF 53364160 Ki = 12 nM T20401 C32UEX 53364161 Ki = 11 nM T20401 CHWX25 53364162 Ki = 85 nM T20401 C58YMC 53371608 Ki = 569 nM T20401 C0NUM6 53386724 Ki = 279 nM T20401 C54FGU 53386866 Ki = 21.5 nM T20401 CRI54V 53386867 Ki = 980 nM T20401 CUX7S4 53386868 Ki = 955 nM T20401 CSA60L 53389267 Ki = 450 nM T20401 C8VXD9 53389268 Ki = 41.3 nM T20401 CV40HR 53426278 Ki = 6.2 nM T20401 CUI84R 53439104 Ki = 30000 nM T20401 C6T5RC 53483944 Ki = 4890 nM T20401 CM5KX6 53483945 Ki = 6315 nM T20401 C3M4EL 53483958 Ki = 4125 nM T20401 CCFP92 53516400 Ki = 5.7 nM T20401 CY2MI0 54077127 Ki > 10000 nM T20401 CXO38A 54444800 IC50 = 165 nM T20401 CB6W4D 54577841 Ki > 10000 nM T20401 CI83DC 54578707 Ki = 42.6 nM T20401 CHCT45 54580732 Ki = 12 nM T20401 CEAP89 54581017 Ki = 96000 nM T20401 CYB47X 54581736 Ki = 14 nM T20401 CJI09P 54582050 Ki = 112000 nM T20401 CW2KI4 54582723 Ki = 10 nM T20401 CWK6B0 54582724 Ki = 71 nM T20401 CXR63W 54583699 Ki = 1.4 nM T20401 CBS8R1 54584666 Ki = 33 nM T20401 CJ3UE2 54584667 Ki = 101 nM T20401 C69YAR 54584941 Ki = 281000 nM T20401 CO0BD9 54585508 Ki = 88 nM T20401 CN1LI2 54592380 Ki = 13 nM T20401 C0A5OZ 54612935 Ki = 4.2 nM T20401 C6SM5T 54613427 Ki = 3130 nM T20401 C6X7QG 54613732 Ki = 0.08 nM T20401 CKB0G9 54669765 Ki = 5.3 nM T20401 CS8IV7 54669781 Ki = 5.5 nM T20401 C0PJ1K 54677403 Ki > 10000 nM T20401 CAS91K 54682930 Ki > 100000 nM T20401 CQ3XK0 54758050 Ki = 11.2 nM T20401 C5ON9E 54758136 Ki = 10.6 nM T20401 C0K2LN 54758137 Ki = 38.5 nM T20401 C5Q9XC 54758138 Ki = 49.8 nM T20401 CLT0W2 54758232 Ki = 44.5 nM T20401 C5V4GI 54758233 Ki = 10.7 nM T20401 C98JVL 54758234 Ki = 49.2 nM T20401 CXBF42 54758235 Ki = 37.9 nM T20401 C4EL5V 54758236 Ki = 59.5 nM T20401 CU19DH 54758322 Ki = 48.2 nM T20401 CE53AN 54758323 Ki = 11.9 nM T20401 CK3Q0O 54758324 Ki = 219 nM T20401 CE2O3A 54768697 Ki = 220 nM T20401 C5SB4M 54768698 Ki = 487 nM T20401 CBNP25 54768699 Ki = 54.6 nM T20401 C9Z4RJ 54772055 Ki = 102 nM T20401 CB3EC8 54772057 Ki = 336 nM T20401 CE6LD4 54772059 Ki = 391 nM T20401 CD5P1I 54772061 Ki = 149 nM T20401 C3RQX8 54940826 Ki = 84.5 nM T20401 C0ZJ2L 55629711 Ki = 6.2 nM T20401 CGR24P 56659114 Ki = 11 nM T20401 CRHT26 56659115 Ki = 6 nM T20401 CD56GS 56659116 Ki = 20 nM T20401 CK89GH 56659335 Ki = 435 nM T20401 C05JRQ 56659336 Ki = 435 nM T20401 CEC29W 56659337 Ki = 409 nM T20401 C2TW1F 56659553 Ki = 9.6 nM T20401 CO9SW8 56659554 Ki = 351 nM T20401 CVRM21 56659555 Ki = 15 nM T20401 CJ43WP 56659826 Ki = 21200 nM T20401 CP5QI2 56662619 Ki = 0.4 nM T20401 CZ4HI1 56662794 Ki = 412 nM T20401 CD8SR3 56662795 Ki = 119 nM T20401 CF0J6I 56663002 Ki = 9.6 nM T20401 CH0MV2 56663442 Ki = 5200 nM T20401 CM07OK 56663443 Ki = 2140 nM T20401 C6M0HP 56666075 Ki = 8 nM T20401 CVM8W4 56666268 Ki = 376 nM T20401 C89SEG 56666269 Ki = 258 nM T20401 C36TYE 56666270 Ki = 517 nM T20401 CD5OZ4 56666482 Ki = 9.7 nM T20401 CI93KS 56666719 Ki = 48500 nM T20401 CKT5V0 56669476 Ki = 9 nM T20401 C9NV7U 56669478 Ki = 0.8 nM T20401 CR9F8U 56670316 Ki = 5290 nM T20401 CF1J7H 56670317 Ki = 4610 nM T20401 CWNF20 56673403 Ki = 295 nM T20401 CT29KP 56673404 Ki = 486 nM T20401 C7DU3M 56673405 Ki = 22.1 nM T20401 CHV04E 56673655 Ki = 82 nM T20401 C4YI1B 56673656 Ki = 4680 nM T20401 CKL09N 56673817 Ki = 1710 nM T20401 C8SY2J 56676310 Ki = 0.8 nM T20401 CI2R9B 56676517 Ki = 368 nM T20401 C9X7VM 56676518 Ki = 561 nM T20401 CF86WB 56676713 Ki = 13.9 nM T20401 CDH07V 56677155 Ki = 5220 nM T20401 CR7D6S 56677156 Ki = 4950 nM T20401 CSKB42 56679637 Ki = 0.7 nM T20401 C2U1VF 56679839 Ki = 453 nM T20401 CS81JH 56680034 Ki = 88 nM T20401 C02WBE 56680461 Ki = 57 nM T20401 C7D2IN 56682958 Ki = 6 nM T20401 CGX98C 56682960 Ki = 0.7 nM T20401 C2UE8F 56682961 Ki = 7 nM T20401 CEZ3F5 56683163 Ki = 356 nM T20401 C4LB1M 56683164 Ki = 475 nM T20401 CZS9V5 56683165 Ki = 371 nM T20401 C8V1PA 56683626 Ki = 76 nM T20401 CXL7Q1 56683627 Ki = 22300 nM T20401 CIJ9V0 56684131 Ki = 49 nM T20401 C6IAC4 56689569 Ki > 50000 nM T20401 CTWZ62 56836370 Ki = 418 nM T20401 C49PBJ 56836371 Ki = 215 nM T20401 CK7Y8J 56836443 Ki = 97.4 nM T20401 CY7Z1A 56836444 Ki = 410 nM T20401 CV0ST7 56836445 Ki = 170 nM T20401 C0O3UI 56836446 Ki = 196 nM T20401 C0PKB5 56836447 Ki = 335 nM T20401 CZ9F7P 56836511 Ki = 0.93 nM T20401 COY29V 56836512 Ki = 58.2 nM T20401 C7PWG1 56836513 Ki = 0.94 nM T20401 C4CF8M 56836514 Ki = 0.97 nM T20401 C4IRK8 56836515 Ki = 362 nM T20401 CH52DA 56921864 Ki = 2010 nM T20401 C0Z8WY 56925533 Ki = 590 nM T20401 CTFL92 56928044 Ki = 8.6 nM T20401 CC3Q9S 56928516 Ki = 74.1 nM T20401 CO18AP 57011620 Ki = 21.4 nM T20401 C4VGE9 57047254 Ki = 9.2 nM T20401 CNG76Q 57326130 Ki = 3.6 nM T20401 C81YCD 57326131 Ki = 33 nM T20401 C4TV1U 57326132 Ki = 29.4 nM T20401 CHL0B3 57326133 Ki = 36.3 nM T20401 C5Z4SW 57326134 Ki = 13.5 nM T20401 CFU62Y 57326227 Ki = 20.3 nM T20401 C97HYX 57326228 Ki = 24.7 nM T20401 CS4I5T 57326229 Ki = 17.3 nM T20401 CUR32K 57334711 Ki = 380 nM T20401 C2CD1R 57334712 Ki = 380 nM T20401 C1K0DM 57334713 Ki = 390 nM T20401 CP7YR5 57345662 Ki > 200000 nM T20401 C0S2YZ 57383964 Ki = 376 nM T20401 C97GHV 57383965 Ki = 271 nM T20401 CXW5D3 57384052 Ki > 100000 nM T20401 C4XF9A 57384114 Ki = 539 nM T20401 CS76WU 57384115 Ki = 377 nM T20401 C0UBL5 57384116 Ki = 525 nM T20401 C16AGY 57384117 Ki = 344 nM T20401 CVWK43 57386884 Ki > 100000 nM T20401 CR3C7D 57386885 Ki > 100000 nM T20401 C9CX4B 57386886 Ki > 100000 nM T20401 CZOD69 57386887 Ki > 200000 nM T20401 CZN72E 57386888 Ki > 100000 nM T20401 C9JU0H 57386889 Ki > 100000 nM T20401 CQ0I4V 57386890 Ki > 200000 nM T20401 C8Z0DJ 57387135 Ki > 200000 nM T20401 C1HZS5 57387136 Ki > 200000 nM T20401 C7EN6Z 57387137 Ki > 200000 nM T20401 C87ASQ 57387395 Ki > 100000 nM T20401 CQW5T3 57387397 Ki > 100000 nM T20401 CT3B0Z 57387636 Ki > 100000 nM T20401 CV4C7B 57390570 Ki = 104 nM T20401 CS5O2D 57390571 Ki = 88 nM T20401 C14VNC 57390572 Ki = 320 nM T20401 C09GQI 57392249 Ki = 7 nM T20401 CY81SU 57392250 Ki = 8.6 nM T20401 CMEV16 57392251 Ki = 9.8 nM T20401 C94YIX 57392252 Ki = 7 nM T20401 CDP3C2 57392352 Ki = 293 nM T20401 C13FJU 57392368 Ki = 410 nM T20401 CM7S3H 57394009 Ki = 10 nM T20401 CHAF57 57394010 Ki = 10.2 nM T20401 CV7K9Y 57394771 Ki = 222 nM T20401 CM4SL9 57394772 Ki = 6.9 nM T20401 C1M0LS 57394809 Ki = 520 nM T20401 CJ5XK2 57395770 Ki = 7.3 nM T20401 CV6QX4 57395771 Ki = 297 nM T20401 CP9D5B 57395861 Ki = 4184 nM T20401 CY5G4Z 57395885 Ki = 840 nM T20401 C5RX6H 57396029 Ki = 4330 nM T20401 CHG91B 57396529 Ki = 9.3 nM T20401 C9H4VS 57396530 Ki = 7.4 nM T20401 C6XD2O 57397549 Ki = 7.3 nM T20401 C64VIW 57397550 Ki = 6.4 nM T20401 CR30XN 57397648 Ki = 91 nM T20401 CP75OF 57397664 Ki = 34560 nM T20401 CUAG84 57397836 Ki = 58910 nM T20401 CW43HV 57397837 Ki = 4420 nM T20401 CRIU35 57398318 Ki = 109 nM T20401 CN6TU2 57398319 Ki = 9 nM T20401 C97OJM 57399231 Ki = 7.8 nM T20401 C7XAZ3 57399232 Ki = 8.7 nM T20401 CK24NA 57399233 Ki = 108 nM T20401 C1MCW8 57399336 Ki = 69120 nM T20401 C2CAM1 57399491 Ki = 3970 nM T20401 CQD65L 57401080 Ki = 476 nM T20401 C1SK7F 57401081 Ki = 222 nM T20401 CG3X4V 57401764 Ki = 105 nM T20401 C4V5KY 57402747 Ki = 524 nM T20401 CRU53E 57402748 Ki = 11.9 nM T20401 C52TUM 57402749 Ki = 7.6 nM T20401 CQ9ZG2 57402750 Ki = 390 nM T20401 C6GO4Q 57402755 Ki = 3 nM T20401 CI3L9R 57402843 Ki = 422 nM T20401 CW10QX 57402844 Ki = 99.7 nM T20401 C80WTZ 57403496 Ki = 60 nM T20401 CDIM87 57403497 Ki = 7.5 nM T20401 C76ZDS 57404539 Ki = 7.4 nM T20401 CKID78 57411990 Ki = 21 nM T20401 C4ZYF3 57411991 Ki = 5.6 nM T20401 CDG6R4 57411992 Ki = 10.1 nM T20401 CKPS17 57411993 Ki = 4.5 nM T20401 CV13LT 57411994 Ki = 361 nM T20401 CW1TU4 57412422 Ki = 33 nM T20401 CT4BV9 57412423 Ki = 5.3 nM T20401 C31NWX 57412424 Ki = 4.9 nM T20401 CD86ER 57412425 Ki = 87.5 nM T20401 CB94YU 57412426 Ki = 8.8 nM T20401 C2K8YJ 57412507 Ki = 8.8 nM T20401 CSF4V6 57412508 Ki = 43.5 nM T20401 CHAO86 57412509 Ki = 8.9 nM T20401 C3U6TH 57412510 Ki = 84.5 nM T20401 C40LOS 57412511 Ki = 48.5 nM T20401 CZ47VT 57412512 Ki = 33.2 nM T20401 C28WRD 57412600 Ki = 86.7 nM T20401 C2XPG5 57413583 Ki = 6.3 nM T20401 CM2AY7 57413584 Ki = 6.7 nM T20401 C5JDQ1 57413825 Ki = 330 nM T20401 C5M4CN 57413826 Ki = 3.8 nM T20401 C3D7KS 57413827 Ki = 37 nM T20401 CJO26X 57413828 Ki = 4.8 nM T20401 CA4CD7 57413968 Ki = 10.1 nM T20401 CQ1ZK6 57519697 Ki = 74 nM T20401 CX8W0C 57624955 IC50 = 530 nM T20401 C3AUH6 57901193 IC50 = 36000 nM T20401 CG3W0D 58404071 Ki = 173 nM T20401 CT3B7P 58477593 Ki = 56.2 nM T20401 C01TQW 59079460 Ki = 11.6 nM T20401 CF1NG0 60155028 Ki = 2.176 nM T20401 C0PRW7 60155029 Ki = 2.17 nM T20401 CNX97Q 60155030 Ki = 2.018 nM T20401 CR0Z7W 60155031 Ki = 2.13 nM T20401 CI2WL7 60155120 Ki = 2.472 nM T20401 CM57BF 60155121 Ki = 2.305 nM T20401 C5VF9X 60155122 Ki = 1.98 nM T20401 C2U8VH 60155123 Ki = 2.092 nM T20401 CNR53M 60155124 Ki = 760 nM T20401 CYQM98 60201413 Ki = 1170 nM T20401 CGWU14 60201414 Ki = 59 nM T20401 C6TP2W 60201415 Ki = 9.1 nM T20401 C1JVP9 60201416 Ki = 178 nM T20401 CQZN79 60201417 Ki = 63 nM T20401 CVU0B4 60201577 Ki = 62 nM T20401 CS3N6M 60201578 Ki = 0.6 nM T20401 CB45GM 60201579 Ki = 5.2 nM T20401 C9V6EY 60446869 Ki = 385.6 nM T20401 COW0X5 61580695 Ki = 236 nM T20401 C1CVG9 61580845 Ki = 110 nM T20401 C9UD2V 62141270 Ki = 2340 nM T20401 CZ4BQ6 66571808 Ki > 10000 nM T20401 CGB46T 66571809 Ki > 10000 nM T20401 CT0S3A 66572208 Ki > 10000 nM T20401 C2J7GW 66572313 Ki = 54430 nM T20401 C7J5RN 66573254 Ki = 78490 nM T20401 CGF3W6 66586679 Ki = 700 nM T20401 CN84CU 66586879 Ki = 580 nM T20401 CAD3V2 67662627 Ki = 181 nM T20401 C54HCL 68341722 Ki = 94.4 nM T20401 C4MB5P 68602550 Ki > 10000 nM T20401 CA7F0J 68819643 Ki = 176 nM T20401 CV6PY2 68833705 Ki = 1.2 nM T20401 CIGB32 68875681 IC50 = 156 nM T20401 C23JZS 70037678 Ki = 341 nM T20401 C6RVC3 70202738 Ki = 8.2 nM T20401 C3BYV1 70681295 IC50 = 36200 nM T20401 CDO92J 70681983 Ki = 2.039 nM T20401 CHC54M 70681984 Ki = 2.177 nM T20401 C1FY3K 70681985 Ki = 2.018 nM T20401 CSW7I0 70681986 Ki = 2.142 nM T20401 CP65RU 70681987 Ki = 1.972 nM T20401 CFT68C 70681988 Ki = 2.097 nM T20401 C2Y5KV 70682044 Ki = 2150 nM T20401 CR0D9S 70684100 Ki = 2.177 nM T20401 CRZ8S1 70684101 Ki = 2.105 nM T20401 COS95H 70684102 Ki = 2.179 nM T20401 CT5PH1 70684103 Ki = 1.846 nM T20401 CK48WR 70684962 IC50 = 44 nM T20401 C4SX6F 70685487 IC50 = 6790 nM T20401 C9P4BK 70685635 Ki = 40.8 nM T20401 C5XTY9 70686245 Ki = 2.009 nM T20401 C5A6TI 70687643 IC50 = 8740 nM T20401 C4SCY0 70688360 Ki = 1.964 nM T20401 CPD1N7 70688361 Ki = 1.752 nM T20401 C4L2OE 70688362 Ki = 1.758 nM T20401 CZO9C5 70688363 Ki = 1.879 nM T20401 CAD39I 70688364 Ki = 2.132 nM T20401 CRHL03 70689373 Ki = 0.4 nM T20401 CVQ6B2 70689703 IC50 = 8250 nM T20401 C9G7QF 70689704 IC50 = 8350 nM T20401 C7N4RT 70690386 Ki = 1.995 nM T20401 CQD8R9 70690387 Ki = 1.982 nM T20401 C1T4JL 70690936 Ki = 4350 nM T20401 CUY3O8 70690937 Ki = 1190 nM T20401 C5C9SL 70691832 IC50 = 13700 nM T20401 CP81SC 70691833 IC50 = 9020 nM T20401 CQR91N 70692438 Ki = 34620 nM T20401 CXF59L 70692549 Ki = 2.364 nM T20401 CV76WB 70692550 Ki = 1.999 nM T20401 C89LCZ 70692551 Ki = 2.159 nM T20401 C1K8VS 70692552 Ki = 1.827 nM T20401 CO5JP7 70692553 Ki = 2.558 nM T20401 CK5Y7G 70692554 Ki = 2.179 nM T20401 CGD06J 70692555 Ki = 1.9 nM T20401 C5QOK4 70692556 Ki = 1.987 nM T20401 CF0YQ6 70693894 IC50 = 8070 nM T20401 C4BDK3 70694601 Ki = 2.35 nM T20401 CW8YA7 70694602 Ki = 1.678 nM T20401 CCYE61 70694603 Ki = 2.093 nM T20401 CEF1J8 70694604 Ki = 1.895 nM T20401 C4C0HK 70694605 Ki = 2.148 nM T20401 CBDQ72 70694606 Ki = 2.261 nM T20401 C95YWO 70695124 Ki = 3620 nM T20401 CSH7P1 70696148 Ki = 27.8 nM T20401 CWJ0Q8 70696540 Ki = 26376 nM T20401 CWSA94 70696638 Ki = 2.149 nM T20401 CREC06 70696639 Ki = 2.188 nM T20401 CJ4M9S 70696640 Ki = 2.18 nM T20401 CHFY23 70696641 Ki = 2.186 nM T20401 C3Z7ER 70696642 Ki = 1.722 nM T20401 C6E4UW 70696643 Ki = 2.092 nM T20401 C0SP9E 70696644 Ki = 1.947 nM T20401 CAFH02 70696645 Ki = 1.992 nM T20401 CWQM13 70696646 Ki = 2.224 nM T20401 CL1Z8G 70697527 IC50 = 7.1 nM T20401 C51HSA 70791252 IC50 = 2800 nM T20401 CNS4U0 70791951 Ki = 439 nM T20401 CS58EL 70792049 Ki = 456 nM T20401 C8FB0P 71273627 Ki = 1.805 nM T20401 CJH6Y7 71273628 Ki = 2.096 nM T20401 CXG0H9 71273629 Ki = 1.994 nM T20401 CUT6R1 71273630 Ki = 1.805 nM T20401 CH49BT 71273631 Ki = 2.019 nM T20401 CK2U8R 71273632 Ki = 2.007 nM T20401 C2F9PC 71273633 Ki = 2.138 nM T20401 CV8FW3 71273635 Ki = 1.682 nM T20401 CQJ61A 71273738 Ki = 2.084 nM T20401 CSMV41 71273739 Ki = 2.503 nM T20401 CYW59B 71273740 Ki = 2.135 nM T20401 CU0KV6 71273743 Ki = 2.469 nM T20401 CC21VR 71273744 Ki = 2.438 nM T20401 C80KUG 71273750 Ki = 2.139 nM T20401 CJHN78 71415156 Ki = 11 nM T20401 C8NYL3 71449075 Ki = 9 nM T20401 CRN2O1 71449118 Ki = 14.7 nM T20401 C16PMU 71449958 IC50 = 9590 nM T20401 CXJ16H 71450117 Ki = 72 nM T20401 CR79UB 71450332 Ki = 620 nM T20401 C09RTJ 71450813 Ki = 18 nM T20401 C6VQI7 71450814 Ki = 14 nM T20401 CK04AG 71450862 Ki = 0.5 nM T20401 CU3XD2 71450931 Ki = 1 nM T20401 C72GOW 71450940 Ki = 48 nM T20401 CT8E7N 71451561 Ki = 49 nM T20401 CHI2Z6 71452138 Ki = 318 nM T20401 CNI0R5 71452603 Ki = 669 nM T20401 C9D3CU 71452683 Ki = 10 nM T20401 CE4HO5 71453463 Ki = 10 nM T20401 C4E6PS 71453593 IC50 = 610 nM T20401 CP27AT 71453970 Ki = 513 nM T20401 CW49YT 71453971 Ki = 404 nM T20401 C52WNJ 71454366 Ki = 453 nM T20401 CT90CD 71454373 Ki = 56.7 nM T20401 CKB14Q 71454522 Ki = 11 nM T20401 CZ0P8A 71454523 Ki = 2 nM T20401 CB8JA3 71455488 Ki = 210 nM T20401 C02UHX 71455489 Ki = 16 nM T20401 CZ0S7D 71455712 Ki = 339 nM T20401 CUX07I 71455715 Ki = 726 nM T20401 C9COK3 71456113 Ki = 873 nM T20401 CICJ97 71457274 Ki = 29 nM T20401 CL2BN6 71457492 Ki = 379 nM T20401 C4L0BG 71457918 Ki = 674 nM T20401 C0XQ5P 71457958 Ki = 15 nM T20401 CSD08X 71458070 Ki = 160 nM T20401 CWHN25 71459359 Ki = 358 nM T20401 CE31LC 71459360 Ki = 700 nM T20401 C7G6IR 71459681 Ki = 49200000 nM T20401 C70MBK 71459826 Ki = 688 nM T20401 C95MKT 71459827 Ki = 573 nM T20401 C5WYI8 71459828 Ki = 461 nM T20401 CX9KJ3 71459903 Ki = 16 nM T20401 CO30KR 71459904 Ki = 23 nM T20401 CJX65D 71459953 Ki = 8 nM T20401 C14NRE 71459973 Ki = 25 nM T20401 CD93TU 71461134 Ki = 568 nM T20401 C3WKX5 71461135 Ki = 567 nM T20401 C3YSR8 71461136 Ki = 457 nM T20401 CS1WI7 71461542 Ki = 389 nM T20401 C7VQ1R 71461543 Ki = 387 nM T20401 C4X1BZ 71462495 IC50 = 8820 nM T20401 CUM2H8 71462868 Ki = 490 nM T20401 CU4N0L 71462869 Ki = 804 nM T20401 C9KZA2 71462872 Ki = 675 nM T20401 CI6V9W 71489159 Ki = 6950 nM T20401 CDQ8Z3 71498310 IC50 = 142.48 nM T20401 CIE7T0 71498311 IC50 = 949.64 nM T20401 CN6K9Q 71498738 IC50 = 239.58 nM T20401 CX6JP1 71498761 IC50 = 276.83 nM T20401 C98SLI 71498762 IC50 = 166.58 nM T20401 CJ2TX7 71498763 IC50 = 908.13 nM T20401 C0QX8S 71498764 IC50 = 20.75 nM T20401 CQPM90 71508409 Ki = 144 nM T20401 C8CH5R 71508458 Ki = 128 nM T20401 CF4RQ9 71508459 Ki = 159 nM T20401 CJ5KW8 71508507 Ki = 126 nM T20401 C0VWD1 71508508 Ki = 197 nM T20401 CHZ93F 71508509 Ki = 111 nM T20401 CLD8G6 71508510 Ki = 136 nM T20401 C58ZQR 71508548 Ki = 95.4 nM T20401 CBP08O 71508550 Ki = 379 nM T20401 CMHG14 71521493 Ki = 3900 nM T20401 CHN53G 71521494 Ki = 7100 nM T20401 CZJ5M6 71521495 Ki = 5500 nM T20401 CFBE53 71521496 Ki = 7800 nM T20401 CME27W 71521497 Ki = 3100 nM T20401 C24XWU 71521575 Ki = 7000 nM T20401 CJF68W 71521576 Ki = 6800 nM T20401 CHL8P3 71522144 Ki = 8890 nM T20401 CEYG83 71522162 Ki > 100000 nM T20401 CZ78YT 71522163 Ki > 100000 nM T20401 C8NAF3 71545047 Ki = 7760 nM T20401 C4H6PD 71545048 Ki = 6330 nM T20401 CQ20AS 71545049 Ki = 9210 nM T20401 CG2CL6 71545050 Ki = 7200 nM T20401 C1MET8 71545051 Ki = 9290 nM T20401 CILC35 71545052 Ki = 9370 nM T20401 CGQ97W 71545216 Ki = 9640 nM T20401 C71UMX 71545217 Ki = 9350 nM T20401 C3KJ6D 71545218 Ki = 7720 nM T20401 C0JNF3 71545219 Ki = 8610 nM T20401 CRJG87 71552329 Ki = 39.81 nM T20401 CXWK92 71552410 Ki = 5.012 nM T20401 CKW1B5 71552411 Ki = 0.631 nM T20401 CH2A6X 71552499 Ki = 39.81 nM T20401 CYS8X6 71552500 Ki = 100 nM T20401 C4X7BQ 71552593 Ki = 50.12 nM T20401 C83YNA 71552594 Ki = 1.259 nM T20401 C3RI7B 71552595 Ki = 50.12 nM T20401 CI25EH 71552664 Ki = 7.943 nM T20401 C8QM9L 71552665 Ki = 7.943 nM T20401 CC5EB7 71570660 Ki = 213.76 nM T20401 CA82YW 71570661 Ki = 1389.5 nM T20401 CNL58G 71570662 Ki = 104.52 nM T20401 CQKG46 71578358 Ki = 8860 nM T20401 CV6FW1 71578359 Ki = 3090 nM T20401 CDA18G 71578360 Ki = 6750 nM T20401 C3P8YG 71578361 Ki = 13440 nM T20401 CDGY15 71578422 Ki = 95.6 nM T20401 CA5M6S 71578423 Ki = 61.7 nM T20401 CGOR42 71578424 Ki = 54.8 nM T20401 C45YXJ 71578425 Ki = 61.7 nM T20401 C1CKL6 71578426 Ki = 28.2 nM T20401 CR38IX 71578427 Ki = 27.1 nM T20401 CQ8Z5T 71578500 Ki = 6.7 nM T20401 CZ1R3F 71578570 Ki = 4.2 nM T20401 CV0G1A 71578571 Ki = 31.3 nM T20401 CX7T2V 71578640 Ki = 7.9 nM T20401 COT80J 71578641 Ki = 43 nM T20401 CGV68Z 71578723 Ki = 122 nM T20401 C7U0LV 71578724 Ki = 237 nM T20401 C8M0YB 71578725 Ki = 153 nM T20401 C4F0HB 71578726 Ki = 46 nM T20401 CZ29IK 71578808 Ki = 9.6 nM T20401 C8HMK5 71578809 Ki = 264 nM T20401 CMH2W4 71578810 Ki = 388 nM T20401 C7W9BS 71578811 Ki = 8.9 nM T20401 CU6N9T 71578812 Ki > 10000 nM T20401 CGEJ87 71578813 Ki = 381 nM T20401 C8CM0Q 71578898 Ki = 490 nM T20401 C19JFD 71578899 Ki = 782 nM T20401 C0MT2F 71578903 Ki = 142 nM T20401 CB9R7F 71578904 Ki = 9.1 nM T20401 C5MLA7 71578977 Ki = 170 nM T20401 C03THE 71578978 Ki = 250 nM T20401 CR57YV 71578979 Ki = 290 nM T20401 CVTN91 71578980 Ki = 57.54 nM T20401 CBJ18U 71578981 Ki = 4708 nM T20401 CCKJ51 71578982 Ki = 75 nM T20401 C0TKR8 71579053 Ki = 5176 nM T20401 CX4D6V 71579054 Ki = 1400 nM T20401 CJ0UP9 71579055 Ki = 85.3 nM T20401 CREN23 71579056 Ki = 799.1 nM T20401 CP61GE 71579057 Ki = 4235 nM T20401 CXD68U 71579058 Ki = 4995 nM T20401 C19OIY 71579130 Ki = 490 nM T20401 CG8X1V 71584198 Ki = 3.5 nM T20401 CV0LU6 71602117 Ki = 510 nM T20401 CCE15B 71602410 Ki = 27.6 nM T20401 CCB72P 71602411 Ki = 9.1 nM T20401 CHL16T 71602412 Ki = 26.2 nM T20401 C2UQV5 71602471 Ki = 6.2 nM T20401 C8K1YM 71602472 Ki = 5.6 nM T20401 CZL96Y 71602476 Ki = 5.2 nM T20401 CE70AQ 71602537 Ki = 238 nM T20401 C3KPA8 71602538 Ki = 47.2 nM T20401 CO6FJ4 71602539 Ki = 8.6 nM T20401 CQ17LM 71602540 Ki = 5.3 nM T20401 C78LKP 71607884 IC50 > 10000 nM T20401 COVC80 71607885 IC50 > 10000 nM T20401 C1MOS8 71607912 IC50 = 61.8 nM T20401 CE0F4T 71607913 IC50 > 10000 nM T20401 CO2LM4 71607914 IC50 > 10000 nM T20401 CNBK57 71607915 IC50 > 10000 nM T20401 CXPO21 71607916 IC50 > 10000 nM T20401 CU24SZ 71607951 IC50 = 26.8 nM T20401 CJQW86 71607952 IC50 = 455.1 nM T20401 CR7BQ5 71607953 IC50 = 146.5 nM T20401 CPM89A 71607954 IC50 > 10000 nM T20401 C1OPS4 71658869 Ki = 2.03 nM T20401 CN2FZ3 71659103 Ki = 2.95 nM T20401 CC0EU9 71677604 Ki = 60.7 nM T20401 CS4VW3 71681364 Ki = 366 nM T20401 C5SY2L 71681517 Ki = 8.1 nM T20401 CT1D0W 71681519 Ki = 9.5 nM T20401 CW65GP 71681521 Ki = 59 nM T20401 CFS62D 71681523 Ki = 5.4 nM T20401 C96OCT 71681525 Ki = 13.1 nM T20401 C57BRD 71681527 Ki = 21.5 nM T20401 CU45ER 71681529 Ki = 6.4 nM T20401 C5DEF6 71714067 Ki = 21800 nM T20401 C50LSJ 71714068 Ki = 36900 nM T20401 C6A1RS 71716868 Ki = 11 nM T20401 C84WSV 71716939 Ki = 2370 nM T20401 CBY8J3 71716994 Ki = 4600 nM T20401 CM4T1R 71717003 Ki > 100000 nM T20401 CN76CQ 71717054 Ki = 36 nM T20401 CI0SY3 71717570 Ki = 800 nM T20401 CYGT30 71717571 Ki = 2030 nM T20401 C7AL0E 71717694 Ki = 11.3 nM T20401 CG4I1X 71718239 Ki = 4700 nM T20401 CUT0L6 71718312 Ki = 11.3 nM T20401 C4N3VH 71718790 Ki = 1.983 nM T20401 C0LYX1 71718858 Ki = 1920 nM T20401 C4B8KN 71718888 Ki = 38 nM T20401 C7U6NR 71719377 Ki > 100000 nM T20401 CM24ND 71719433 Ki = 530 nM T20401 CT3D5S 71719441 Ki = 4400 nM T20401 CY3CV6 71719496 Ki = 31 nM T20401 CJG34A 71720036 Ki = 78900 nM T20401 CIU4L2 71720670 Ki = 6800 nM T20401 CN0L8Q 71720672 Ki = 431 nM T20401 CY54DH 71728127 Ki = 2.5 nM T20401 C9JAE7 71728128 Ki = 1.5 nM T20401 C6HOP3 71728129 Ki = 1.5 nM T20401 CRY5D8 71728130 Ki = 2.2 nM T20401 CM91JE 71728236 Ki = 3.4 nM T20401 C30ZEI 71728237 Ki = 2.2 nM T20401 C4JB8W 71728238 Ki = 2.6 nM T20401 C5RS9P 71728239 Ki = 1.9 nM T20401 CRYC54 71728240 Ki = 1.8 nM T20401 CLI52C 71732474 IC50 > 10000 nM T20401 C5TKY7 71764398 Ki = 0.96 nM T20401 CMD91U 71764399 Ki = 8.7 nM T20401 CXO1T9 71764400 Ki = 6.9 nM T20401 CVEI80 71764401 Ki = 1.9 nM T20401 CVQ1H3 71764402 Ki = 0.78 nM T20401 CRZ64M 71764403 Ki = 9.5 nM T20401 CC0X1H 71764607 Ki = 7.3 nM T20401 CK7NI0 71764608 Ki = 0.91 nM T20401 C90YMG 71764609 Ki = 0.74 nM T20401 CK35HL 71764610 Ki = 8.9 nM T20401 C4SV1I 71764611 Ki = 0.94 nM T20401 C8NG9B 71764612 Ki = 0.8 nM T20401 CA2M1B 71764613 Ki = 0.69 nM T20401 CR7J6M 71764825 Ki = 0.77 nM T20401 CG09CJ 71764826 Ki = 0.72 nM T20401 CK2N0Z 71764827 Ki = 3.2 nM T20401 C08RAW 71765040 Ki = 0.7 nM T20401 CGI1J3 71765041 Ki = 0.7 nM T20401 CPT1X2 71765042 Ki = 0.76 nM T20401 CHC9K2 71768354 Ki = 11 nM T20401 C0ROQ1 71770179 Ki = 2.9 nM T20401 C8W6DJ 71770180 Ki = 27.7 nM T20401 CB3Y0X 71770181 Ki = 4515 nM T20401 CKHM42 71770182 Ki = 3.4 nM T20401 CBL41T 71770183 Ki = 4.9 nM T20401 C30EYH 71770184 Ki = 2.4 nM T20401 CGA62Y 71770789 Ki = 6.1 nM T20401 C8GP3J 71770790 Ki = 3.8 nM T20401 C04WFV 71770791 Ki = 3.5 nM T20401 CN4QC0 71770911 Ki = 2.9 nM T20401 C6XSA1 71770912 Ki = 6.3 nM T20401 C5YU4I 71770913 Ki = 2.4 nM T20401 C4G3HO 71770914 Ki = 2.9 nM T20401 CSU93P 71770915 Ki = 7.7 nM T20401 C9NAK1 71770916 Ki = 4.5 nM T20401 C42KOE 71770917 Ki = 3.2 nM T20401 CE8IC7 71770918 Ki = 3 nM T20401 CQJI19 71771031 Ki = 2.7 nM T20401 C2ZOB7 71771032 Ki = 2.9 nM T20401 C93LEJ 71771033 Ki = 2.7 nM T20401 C5UZM3 71771034 Ki = 2.2 nM T20401 CX9N5F 71818212 Ki > 10000 nM T20401 C5IU0Y 72163201 Ki = 68 nM T20401 CNP42E 72163326 Ki = 21 nM T20401 C2KE5D 72163327 Ki = 47 nM T20401 C0Q5XL 72163343 Ki = 71 nM T20401 C63MIX 72163344 Ki = 80 nM T20401 CL3WV2 72163345 Ki = 79 nM T20401 C4T9DA 72163346 Ki = 190 nM T20401 CTK07O 72163347 Ki = 96 nM T20401 CE32BF 72163348 Ki = 55 nM T20401 CBN48K 72163465 Ki = 15 nM T20401 CGB02D 72163466 Ki = 29 nM T20401 CVFN85 72163467 Ki = 23 nM T20401 C82RDA 72163468 Ki = 41 nM T20401 CA1X6Z 72163476 Ki = 47 nM T20401 C7TKJ4 72163610 Ki = 23 nM T20401 C70OBD 72163611 Ki = 46 nM T20401 CA0Q4T 72163612 Ki = 49 nM T20401 C96GMR 72163613 Ki = 65 nM T20401 CJ2K8R 72163743 Ki = 96 nM T20401 CPY81U 72163744 Ki = 59 nM T20401 CC1D3Y 72163745 Ki = 51 nM T20401 CYH0G5 72163746 Ki = 23 nM T20401 CEZM40 72163861 Ki = 33 nM T20401 CMBR85 72163862 Ki = 38 nM T20401 CZ9IE5 72163863 Ki = 67 nM T20401 CZM75P 72163975 Ki = 53 nM T20401 CPT0C9 72163976 Ki = 30 nM T20401 C0FM1E 72202020 Ki = 1.47 nM T20401 CT41SJ 72202021 Ki = 2.04 nM T20401 C12SEI 72203721 IC50 = 33 nM T20401 CR37YX 72203722 IC50 = 58 nM T20401 C4VS2P 72203723 IC50 = 85 nM T20401 CSFR32 72203724 IC50 = 23 nM T20401 CDC0A4 72203725 IC50 = 26 nM T20401 CHUS18 72203726 IC50 = 51 nM T20401 C75RNW 72203906 IC50 = 112 nM T20401 C9AJ0V 72203907 IC50 = 122 nM T20401 C70JFO 72203908 IC50 = 103 nM T20401 CYKE59 72203909 IC50 = 173 nM T20401 CC1SO2 72203951 Ki = 35.4 nM T20401 CE9Q6G 72203952 Ki = 45.2 nM T20401 C5YJK2 72203953 Ki = 33.1 nM T20401 CCGB04 72204081 IC50 = 63 nM T20401 CR8I0V 72204082 IC50 = 88 nM T20401 C6X9ZV 72204083 IC50 = 121 nM T20401 CI5BS4 72204084 IC50 = 100 nM T20401 C72IXW 72204085 IC50 = 141 nM T20401 C3L1TY 72204086 IC50 = 217 nM T20401 CM2F7D 72204122 Ki = 135.5 nM T20401 C8XDF6 72204123 Ki = 38.7 nM T20401 CO51BD 72204124 Ki = 31.8 nM T20401 CWJE09 72204125 Ki = 121.6 nM T20401 C8XVK1 72204126 Ki = 28.4 nM T20401 CL54HN 72204268 IC50 = 173 nM T20401 CQ7U9H 72204269 IC50 = 61 nM T20401 C7WDI2 72204321 Ki > 10000 nM T20401 CX4G0R 72204928 IC50 > 10000 nM T20401 CG9C6U 72204929 IC50 > 10000 nM T20401 C5A6XZ 72204930 IC50 > 10000 nM T20401 C0XZK4 72204931 IC50 > 10000 nM T20401 C6RY4X 72204933 IC50 = 8199 nM T20401 C4N5AB 72204934 IC50 > 10000 nM T20401 C3H2FZ 72205111 IC50 > 10000 nM T20401 CQ0VX7 72205112 IC50 > 10000 nM T20401 CQ7TI1 72205113 IC50 > 10000 nM T20401 CPAW52 72205114 IC50 = 9371 nM T20401 C2LD3J 72205115 IC50 = 7469 nM T20401 C4E2VS 72543811 Ki > 10000 nM T20401 C3UJ8A 72695827 Ki = 5.5 nM T20401 CX82JD 72696463 Ki = 4.9 nM T20401 COCV73 72696591 Ki = 7.1 nM T20401 C5KHD7 72696592 Ki = 5.5 nM T20401 C4FBA6 72696593 Ki = 5.4 nM T20401 CO1JM5 72696594 Ki = 5.6 nM T20401 CUF61Q 72696595 Ki = 5 nM T20401 CB0D5L 72696999 Ki = 167 nM T20401 C1SU0Q 72712917 Ki = 33.8 nM T20401 COD5F4 72712918 Ki = 58 nM T20401 CJW7K4 72712919 Ki > 20000 nM T20401 CT2J8A 72712920 Ki > 20000 nM T20401 CRGC51 72713105 Ki = 52 nM T20401 C61VGR 72713106 Ki = 5.5 nM T20401 C96WHB 72713107 Ki = 2.9 nM T20401 CHPN94 72713108 Ki = 6.6 nM T20401 C8F5CO 72737580 IC50 = 77000 nM T20401 CIO7A1 72737581 IC50 = 220000 nM T20401 C0X2RT 72737582 IC50 = 56000 nM T20401 CRD5N1 72737583 IC50 = 70000 nM T20401 CO5EU7 72737584 IC50 = 75000 nM T20401 C9O1RA 72737585 IC50 = 36000 nM T20401 CT8DN7 72737586 IC50 = 300000 nM T20401 CJB8R7 72792832 Ki = 71.1 nM T20401 C5F7DT 72792833 Ki = 76.3 nM T20401 CAC7J8 72792834 Ki = 573 nM T20401 CFS02B 72792835 Ki = 440 nM T20401 CF5LW1 72792901 Ki = 621 nM T20401 C42IFJ 72792902 Ki = 261 nM T20401 CRMF25 72792903 Ki = 79.4 nM T20401 C2G5SR 72792904 Ki = 181 nM T20401 C6DR9O 72792905 Ki = 174 nM T20401 CGF5O1 72792967 Ki = 661 nM T20401 CWH3N9 72792968 Ki = 8.1 nM T20401 C5DSF8 72792969 Ki = 6.9 nM T20401 C2K6UZ 72792970 Ki = 73.6 nM T20401 CGI8K5 72793036 Ki = 37.9 nM T20401 C8WO6Z 72793037 Ki = 69.1 nM T20401 C6OZ0L 72793038 Ki = 421 nM T20401 CDTQ64 72793039 Ki = 253 nM T20401 CY16FM 72793040 Ki = 6.3 nM T20401 CXQN80 72793101 Ki = 8 nM T20401 CJ19BH 72793102 Ki = 4781 nM T20401 CO1JT3 73054728 Ki = 21 nM T20401 CA2YM5 73056157 Ki = 17.1 nM T20401 CXBJ69 73056158 Ki = 6.4 nM T20401 CT62PI 73056159 Ki = 3.1 nM T20401 CL8V1X 73056160 Ki = 0.94 nM T20401 CX5ZV7 73056161 Ki = 5.8 nM T20401 C1YLW5 73056162 Ki = 0.57 nM T20401 CL1H0W 73056449 Ki = 1.1 nM T20401 C0VNX8 73056450 Ki = 0.89 nM T20401 C8Z6YK 73056451 Ki = 8.6 nM T20401 C0RZW2 73056452 Ki = 0.97 nM T20401 CR2HU6 73056453 Ki = 0.55 nM T20401 CI12KH 73056454 Ki = 4.5 nM T20401 CXHE13 73056743 Ki = 1 nM T20401 C3CHO7 73056744 Ki = 0.93 nM T20401 C3FU9P 73056745 Ki = 4.2 nM T20401 C1G8YT 73056746 Ki = 5.4 nM T20401 CT2S3D 73056747 Ki = 0.91 nM T20401 CM12LF 73056748 Ki = 0.56 nM T20401 C4MIP9 73345840 Ki = 60.4 nM T20401 C4Z7PY 73346473 Ki = 85.3 nM T20401 C48AKL 73346474 Ki = 477 nM T20401 CY2AH8 73346475 Ki = 115 nM T20401 C8QJU7 73346691 Ki = 5.5 nM T20401 C0PA8K 73346692 Ki = 3.6 nM T20401 CT6C3G 73346693 Ki = 2.7 nM T20401 CVN4A3 73346695 Ki = 5.3 nM T20401 CM9K3D 73346697 Ki = 7.8 nM T20401 C3Y4VZ 73347324 Ki = 11.3 nM T20401 C1WQ0C 73347968 Ki = 349 nM T20401 CEHI16 73348197 Ki = 18 nM T20401 C18GUI 73348198 Ki > 1000 nM T20401 C3CJ0F 73349055 Ki = 2.3 nM T20401 C75IEZ 73349056 Ki = 2 nM T20401 CK7MD1 73349516 Ki = 134 nM T20401 CJRE74 73349517 Ki = 87.1 nM T20401 CK98JL 73349518 Ki = 629 nM T20401 C6S7RY 73349758 Ki = 3.2 nM T20401 C2JP5U 73349759 Ki = 370.02 nM T20401 CBL42E 73350409 Ki = 7.8 nM T20401 CP3E7Q 73350410 Ki = 5.1 nM T20401 C38QDY 73351066 Ki = 61.4 nM T20401 COM17Y 73351067 Ki = 295 nM T20401 CN96PE 73351280 Ki = 14 nM T20401 CX1J7D 73352124 Ki = 1.6 nM T20401 CXJL10 73352125 Ki = 2.1 nM T20401 CBN25I 73352538 Ki = 128 nM T20401 CRDB68 73352539 Ki = 389 nM T20401 C4SNT8 73352540 Ki = 1238 nM T20401 C3M2UH 73354029 Ki = 215 nM T20401 C8V2KX 73354879 Ki = 274 nM T20401 CB7Z2K 73355560 Ki = 58.5 nM T20401 CR81ON 73355561 Ki = 76.3 nM T20401 C60FZE 73355562 Ki = 354 nM T20401 CAK9J2 73355834 Ki = 4.9 nM T20401 CC2P6U 73356651 Ki = 7.6 nM T20401 CC9AE6 73356652 Ki = 8.4 nM T20401 C3SB2W 73357104 Ki = 436 nM T20401 C79KVE 73357105 Ki = 96.1 nM T20401 COP7H8 73357339 Ki = 1.9 nM T20401 CA3YT9 73894059 Ki = 21.2 nM T20401 C53JCV 74766009 Ki = 35 nM T20401 C53PBO 74766010 Ki = 19.1 nM T20401 CLPY57 74766011 Ki = 40.3 nM T20401 C7EF5V 76310135 Ki = 87 nM T20401 CLX6H0 76310136 Ki = 89 nM T20401 C9K6XP 76310137 Ki = 15 nM T20401 CX0Y6K 76310141 Ki = 4500 nM T20401 C54AJY 76310148 Ki = 8.5 nM T20401 CR56JE 76310328 Ki > 100000 nM T20401 CCD80R 76310490 Ki > 10000 nM T20401 CUB9V2 76310833 Ki = 390 nM T20401 C4S3QC 76310834 Ki = 831 nM T20401 CY7AV1 76310835 Ki = 31 nM T20401 CTJ50C 76310908 Ki > 50000 nM T20401 CEWJ18 76310909 Ki = 41.4 nM T20401 CR9G4Q 76311013 Ki = 244 nM T20401 CE7O5U 76311014 Ki = 321 nM T20401 CV19YL 76311015 Ki = 325 nM T20401 CO0PZ4 76311101 Ki > 10000 nM T20401 CGT0J3 76311102 Ki > 10000 nM T20401 CD3LU2 76311370 Ki = 53 nM T20401 C3JCD1 76311371 Ki = 230 nM T20401 C70UYF 76311372 Ki = 18 nM T20401 C3JFR9 76311373 Ki = 0.6 nM T20401 C5POS7 76311374 Ki = 56 nM T20401 CI64FZ 76311402 Ki = 80 nM T20401 CVW59F 76311403 Ki = 70 nM T20401 C5RAC6 76311404 Ki = 4.8 nM T20401 CY0R8X 76311405 Ki = 21 nM T20401 C7SO0T 76311406 Ki = 82 nM T20401 CYQ7B0 76311407 Ki = 80 nM T20401 CDGN83 76311408 Ki = 2 nM T20401 C4S6CE 76311409 Ki = 0.7 nM T20401 CTJ63S 76311410 Ki = 0.8 nM T20401 CEW21K 76311421 Ki = 41 nM T20401 C96NRT 76311425 Ki = 48 nM T20401 CG2JI0 76313836 Ki = 23 nM T20401 CD1A5Y 76313837 Ki = 7.8 nM T20401 CU48XE 76313838 Ki = 541 nM T20401 C04EFJ 76313840 Ki = 651 nM T20401 CZ60NF 76313841 Ki = 1359 nM T20401 C5S3XY 76313842 Ki = 3290 nM T20401 CK2LR8 76313848 Ki = 26 nM T20401 CI3WQ5 76313849 Ki = 21 nM T20401 CB2YP3 76313998 Ki = 847 nM T20401 C0KVD7 76314143 Ki > 10000 nM T20401 CE1H8W 76314144 Ki > 10000 nM T20401 C5EM0L 76314145 Ki > 10000 nM T20401 C0T8HW 76314452 Ki = 3780 nM T20401 CZ0JC7 76314453 Ki = 20 nM T20401 CC1Z6A 76314549 Ki = 460 nM T20401 CA1F9S 76314550 Ki > 50000 nM T20401 CZBG52 76314647 Ki = 9.5 nM T20401 C4F7WP 76314648 Ki = 560 nM T20401 C95DKS 76314709 Ki > 10000 nM T20401 C37XBL 76314710 Ki > 10000 nM T20401 C2H7ZA 76314711 Ki > 10000 nM T20401 CE1BX4 76314958 Ki = 270 nM T20401 C9R2KH 76314959 Ki = 71 nM T20401 C1S9BI 76314960 Ki = 1.1 nM T20401 CRO70P 76314961 Ki = 6.5 nM T20401 C06NML 76314962 Ki = 34 nM T20401 C81HKS 76314963 Ki = 210 nM T20401 CY9J1C 76314964 Ki = 75 nM T20401 C9W7DT 76314988 Ki = 5 nM T20401 C5JFN2 76314989 Ki = 98 nM T20401 CKRF91 76314990 Ki = 13 nM T20401 C3C4PI 76315011 Ki = 210 nM T20401 C20MYC 76315012 Ki = 86 nM T20401 C34MRW 76317361 Ki = 156 nM T20401 CXZU92 76317371 Ki = 249 nM T20401 CL5CF8 76317538 Ki > 100000 nM T20401 CB1VD3 76317966 Ki = 54.3 nM T20401 C6GOE1 76318042 Ki = 6.6 nM T20401 CGQ67N 76318218 Ki = 64 nM T20401 CLC1H8 76318279 Ki > 10000 nM T20401 CT7G2Z 76318280 Ki > 10000 nM T20401 CCO80M 76318281 Ki > 10000 nM T20401 CY5O9B 76318282 Ki > 10000 nM T20401 CM5IV7 76318283 Ki > 10000 nM T20401 C4DMY8 76318284 Ki > 10000 nM T20401 CG8QV5 76318285 Ki > 10000 nM T20401 CO18PL 76318590 Ki = 29 nM T20401 C98SVG 76318591 Ki = 32 nM T20401 CH14IG 76318592 Ki = 0.5 nM T20401 CYXT21 76318593 Ki = 1.2 nM T20401 C4J9XP 76318594 Ki = 9 nM T20401 CW59AZ 76318595 Ki = 11 nM T20401 COY1X4 76318596 Ki = 0.6 nM T20401 CU3R6B 76318626 Ki = 310 nM T20401 CT94VN 76318627 Ki = 157 nM T20401 CX2D4V 76318628 Ki = 12 nM T20401 C8SZQ7 76318648 Ki = 21 nM T20401 CFX3A2 76318651 Ki = 13 nM T20401 C1DC8O 76318659 Ki = 52 nM T20401 CDGH94 76321081 Ki = 55 nM T20401 CQ5B4S 76321082 Ki = 349 nM T20401 C9U3LR 76321089 Ki = 3219 nM T20401 CZ2RY8 76321096 Ki = 54 nM T20401 CJM27E 76321273 Ki = 733 nM T20401 C9AP8I 76321274 Ki = 3810 nM T20401 C82NGW 76321408 Ki = 1.7 nM T20401 CWM9C3 76321409 Ki = 887 nM T20401 C78KRT 76321425 Ki > 10000 nM T20401 CJ20ZB 76321688 Ki = 75.9 nM T20401 CVT3O8 76321689 Ki = 67.1 nM T20401 CH36SX 76321755 Ki = 223 nM T20401 C8SZN7 76321756 Ki = 3615 nM T20401 CP24WC 76321814 Ki > 10000 nM T20401 CNP1B7 76321907 Ki = 9.2 nM T20401 C4YP7A 76321908 Ki = 185 nM T20401 CZ31AU 76322240 Ki = 186 nM T20401 C0GF7P 76322242 Ki = 90 nM T20401 CQ5Z3H 76322243 Ki = 50 nM T20401 CIS24L 76322244 Ki = 77 nM T20401 CJN27S 76322270 Ki = 50 nM T20401 C63TZU 76322272 Ki = 120 nM T20401 C4T0DK 76322273 Ki = 81 nM T20401 CYZO10 76322274 Ki = 4.1 nM T20401 C1KL6D 76322275 Ki = 2.8 nM T20401 C7QUH8 76322276 Ki = 10 nM T20401 C1YDG3 76322277 Ki = 9 nM T20401 CG37HT 76322303 Ki = 295 nM T20401 CZ98LC 76324732 Ki = 12 nM T20401 CW87DO 76324733 Ki = 423 nM T20401 C5JXE8 76324738 Ki = 513 nM T20401 CUG2O8 76324739 Ki = 416 nM T20401 CLN0I8 76325020 Ki > 10000 nM T20401 C35EUT 76325021 Ki > 10000 nM T20401 CZQ93S 76325300 Ki = 21.9 nM T20401 CP3X6L 76325374 Ki = 37 nM T20401 CO79TZ 76325375 Ki = 158 nM T20401 CE1DM0 76325376 Ki = 73 nM T20401 CE3P4W 76325377 Ki = 6750 nM T20401 C7ZJ9M 76325378 Ki = 24 nM T20401 CN6CY7 76325452 Ki > 50000 nM T20401 CUC3M2 76325547 Ki = 312 nM T20401 C1BC4A 76325548 Ki = 9.3 nM T20401 CQUE95 76325602 Ki > 10000 nM T20401 CDO73V 76325603 Ki > 10000 nM T20401 C95MSJ 76325864 Ki = 210 nM T20401 C73WKZ 76325865 Ki = 50 nM T20401 CB28DH 76325866 Ki = 14 nM T20401 CV0TP6 76325867 Ki = 55 nM T20401 C68YJL 76325868 Ki = 10 nM T20401 CMRD93 76325869 Ki = 3 nM T20401 C98JBS 76325870 Ki = 275 nM T20401 CE5N1J 76325871 Ki = 17 nM T20401 CL0XR7 76325899 Ki = 0.9 nM T20401 CLI14U 76325900 Ki = 47 nM T20401 C7FI3X 76325901 Ki = 58 nM T20401 C27YJP 76325902 Ki = 42 nM T20401 C4KG1E 76325903 Ki = 210 nM T20401 C4T0VX 76325904 Ki = 170 nM T20401 CO14TP 76325929 Ki = 4 nM T20401 C9F1ZI 76325930 Ki = 0.8 nM T20401 CWP61T 76325931 Ki = 2 nM T20401 C0UK2H 76328279 Ki = 61 nM T20401 CCNB68 76328280 Ki = 985 nM T20401 C8AS9R 76328281 Ki = 357 nM T20401 C3D2QL 76328449 Ki = 47300 nM T20401 CI47ZC 76328450 Ki = 94500 nM T20401 CM05DY 76328451 Ki = 808 nM T20401 CN0KZ1 76328452 Ki = 257 nM T20401 C0CFZ1 76328574 Ki = 34 nM T20401 CYM2G9 76328575 Ki = 3.9 nM T20401 CZ5X4W 76328576 Ki = 140 nM T20401 CP3CN4 76328593 Ki > 10000 nM T20401 CPJM79 76328853 Ki = 72.6 nM T20401 C6F4LU 76328915 Ki = 93 nM T20401 C5VW9J 76328916 Ki = 6585 nM T20401 CEZ6A8 76328917 Ki = 885 nM T20401 CYD50A 76329098 Ki = 178 nM T20401 CB23PR 76329099 Ki = 240 nM T20401 C3QI6J 76329100 Ki = 34 nM T20401 CTF2G1 76329169 Ki > 10000 nM T20401 CAE23D 76329170 Ki > 10000 nM T20401 CX8Z5D 76329449 Ki = 55 nM T20401 CUHX10 76329450 Ki = 218 nM T20401 CU42FB 76329451 Ki = 21 nM T20401 CC69YL 76329452 Ki = 80 nM T20401 C0HJ4Y 76329453 Ki = 106 nM T20401 C3MO2T 76329454 Ki = 71 nM T20401 CEG87T 76329456 Ki = 106 nM T20401 C7WV9M 76329457 Ki = 9 nM T20401 CVWR30 76329482 Ki = 15 nM T20401 CK5S6A 76329483 Ki = 17 nM T20401 CQ85UG 76329484 Ki = 260 nM T20401 CPB5U8 76329485 Ki = 6.1 nM T20401 C6P5UM 76329498 Ki = 280 nM T20401 C6H4KZ 76329499 Ki = 86 nM T20401 CKH0X7 76331969 Ki = 62 nM T20401 CO82ZX 76331970 Ki = 29 nM T20401 C5U7JI 76331976 Ki = 2768 nM T20401 CYC39A 76331984 Ki = 49 nM T20401 CK73VH 76331985 Ki = 146 nM T20401 C5HRL1 76332129 Ki = 27900 nM T20401 C68DOK 76332270 Ki > 10000 nM T20401 CJN0W8 76332271 Ki > 10000 nM T20401 C3ZGF1 76332272 Ki > 10000 nM T20401 C6ENW5 76332521 Ki = 18.3 nM T20401 C4RPU5 76332522 Ki = 40.7 nM T20401 C14UQS 76332523 Ki = 130 nM T20401 CGLB34 76332602 Ki = 5.6 nM T20401 CP9SU7 76332603 Ki = 8760 nM T20401 CG3U6D 76332757 Ki = 71 nM T20401 CSN84K 76332758 Ki = 4 nM T20401 COZ89H 76332830 Ki > 10000 nM T20401 CFI5K7 76332831 Ki > 10000 nM T20401 C5VN9Q 76332832 Ki > 10000 nM T20401 CG9HO7 76333094 Ki = 10 nM T20401 CNB7Q0 76333095 Ki = 240 nM T20401 CNJF36 76333096 Ki = 20 nM T20401 CN1JW9 76333097 Ki = 2.1 nM T20401 CXA5T0 76333098 Ki = 31 nM T20401 CG60RB 76333099 Ki = 50 nM T20401 CJZM43 76333100 Ki = 35 nM T20401 C3K8WP 76333101 Ki = 1.4 nM T20401 CQRM32 76333124 Ki = 96 nM T20401 CDY7R8 76333125 Ki = 156 nM T20401 C8MYW5 76333126 Ki = 315 nM T20401 CEP14I 76333127 Ki = 1.3 nM T20401 C9H4OK 76333128 Ki = 47 nM T20401 CH0YG6 76333129 Ki = 54 nM T20401 C98APF 76333130 Ki = 13 nM T20401 CNH71G 76333131 Ki = 50 nM T20401 C3NQY6 76333149 Ki = 97 nM T20401 CVS5Z9 76333154 Ki = 245 nM T20401 C9W0HZ 76335546 Ki = 98 nM T20401 CZC97G 76335551 Ki = 567 nM T20401 CK5I4M 76335747 Ki = 297 nM T20401 CQKW51 76335889 Ki > 10000 nM T20401 CB53XC 76335911 Ki > 10000 nM T20401 CP16NU 76336199 Ki = 44 nM T20401 C3P4ZB 76336200 Ki = 6.7 nM T20401 CLB17E 76336381 Ki = 579 nM T20401 CV1B6C 76336382 Ki = 681 nM T20401 CWFY73 76336452 Ki > 10000 nM T20401 C2QC4D 76336453 Ki > 10000 nM T20401 CF1PD0 76336721 Ki = 78 nM T20401 CS7E0I 76336722 Ki = 26 nM T20401 C5RLH3 76336723 Ki = 5.6 nM T20401 CXM1A2 76336724 Ki = 180 nM T20401 CO29MN 76336726 Ki = 2.1 nM T20401 CZ78TW 76336727 Ki = 280 nM T20401 CT9V4M 76336730 Ki = 5.2 nM T20401 C0VCW9 76336761 Ki = 0.6 nM T20401 CO21QC 76336762 Ki = 21 nM T20401 C4JB8L 76336763 Ki = 92 nM T20401 CAN2Y3 76336778 Ki = 10 nM T20401 CM67SN 76336780 Ki = 77 nM T20401 CMV08B 76336782 Ki = 62 nM T20401 C5SEZ2 76336785 Ki = 11 nM T20401 CH0OY6 78319159 Ki = 826 nM T20401 CC4F0A 78319160 Ki = 62.1 nM T20401 CO4IE9 78319161 Ki = 772 nM T20401 CY6LN4 78319162 Ki = 8 nM T20401 CU9I6V 82078731 Ki = 140.1 nM T20401 C5TB6O 82080973 Ki = 763.5 nM T20401 CX5WB9 82198349 Ki = 168 nM T20401 C6UZR9 82911195 Ki = 28.7 nM T20401 CVD64Q 83379931 Ki > 10000 nM T20401 CR47YB 86047482 Ki = 49.5 nM T20401 C0P3OF 86047486 Ki = 51.2 nM T20401 CZ5HA6 86047495 Ki = 56.9 nM T20401 CTD2Y9 86276273 Ki = 375 nM T20401 CHY2O4 86276274 Ki = 351 nM T20401 CN7HU3 86288843 Ki = 918 nM T20401 C5Y1WO 86288855 Ki = 703 nM T20401 C76RBA 86298624 IC50 = 504 nM T20401 C93FKI 86298625 IC50 = 70 nM T20401 CVLU48 86298626 IC50 = 71 nM T20401 CR97VD 86692717 Ki = 5.7 nM T20401 C8PC3U 86692718 Ki = 5.2 nM T20401 C6HC8V 86692720 Ki = 5.8 nM T20401 CQ30FJ 86719933 Ki > 100000 nM T20401 C8H6LJ 86765116 IC50 = 129 nM T20401 CH2X9D 88314331 Ki > 10000 nM T20401 C3EYT4 88314336 Ki > 10000 nM T20401 CB4KI9 88973647 Ki = 1625 nM T20401 C1O5YX 90180909 Ki > 100000 nM T20401 CIJ96H 90644155 IC50 > 10000 nM T20401 CX7EW1 90644156 IC50 > 10000 nM T20401 CK5GZ4 90644157 IC50 > 10000 nM T20401 C7O1YN 90644158 IC50 > 10000 nM T20401 CEN6C1 90644159 IC50 = 1830 nM T20401 C8X9UZ 90644160 IC50 = 3820 nM T20401 C6I9RG 90644374 IC50 = 3820 nM T20401 C1DT9W 90644375 Ki = 2680 nM T20401 C2PXK3 90644376 IC50 = 3220 nM T20401 C7OJM0 90644377 Ki = 2510 nM T20401 C3Z8QO 90644378 Ki = 3060 nM T20401 C4QT6W 90644479 Ki = 6.9 nM T20401 C6XB9R 90644480 Ki = 57 nM T20401 C1KXA0 90644481 Ki = 40 nM T20401 C1ND2E 90644482 Ki = 79 nM T20401 CY4LZ9 90644483 Ki = 84 nM T20401 C2RQD9 90644484 Ki = 115 nM T20401 CZ0R6T 90644485 Ki = 164 nM T20401 C4G1BD 90644486 Ki = 123 nM T20401 CL7I9M 90644487 Ki = 87 nM T20401 CVMU79 90644488 Ki = 63 nM T20401 C6F5ZP 90644489 Ki = 13.5 nM T20401 CG85NB 90644490 Ki = 24 nM T20401 CCID31 90644491 Ki = 10.1 nM T20401 C3BPF8 90644492 Ki = 25 nM T20401 C7B5YR 90644493 Ki = 13.1 nM T20401 C9FCX5 90644494 Ki = 8.7 nM T20401 CQND72 90644495 Ki = 47 nM T20401 C4V9IZ 90644496 Ki = 54 nM T20401 C49VLZ 90644497 Ki = 41 nM T20401 CX2I9G 90644498 Ki = 33 nM T20401 C5MXJ4 90644499 Ki = 28 nM T20401 C2E7QM 90644500 Ki = 15.1 nM T20401 CR02MV 90644501 Ki = 29 nM T20401 C2SZ5P 90644502 Ki = 68 nM T20401 C86NMC 90644503 Ki = 44 nM T20401 C8W3PI 90644504 Ki = 39 nM T20401 CF12MK 90645415 Ki = 4.6 nM T20401 CJO6I7 90645416 Ki = 3.2 nM T20401 CU2K5R 90645417 Ki = 3.8 nM T20401 C58KIU 90645418 Ki = 4.9 nM T20401 CS0OX7 90645419 Ki = 4.7 nM T20401 CWD6P7 90645420 Ki = 24.5 nM T20401 CVY5P9 90645421 Ki = 123.7 nM T20401 CAL9C4 90645422 Ki = 4.5 nM T20401 C2EA9C 90645423 Ki = 5.3 nM T20401 C1FVA8 90645424 Ki = 4.9 nM T20401 CP27AX 90645425 Ki = 64.3 nM T20401 C8E4ZH 90645426 Ki = 18.2 nM T20401 C3SIA9 90645429 Ki = 8.5 nM T20401 C1E4FS 90645430 Ki = 5.6 nM T20401 COBQ09 90645431 Ki = 3.9 nM T20401 C7IU8K 90645432 Ki = 7.1 nM T20401 CW0L1D 90654798 Ki = 492 nM T20401 CO2CU1 90654800 Ki = 719 nM T20401 CE54MK 90654802 Ki = 667 nM T20401 CID9U2 90654804 Ki = 6.3 nM T20401 C27QHW 90654822 Ki = 8058 nM T20401 C96OWE 90654823 Ki = 9315 nM T20401 CZQ9E3 90654824 Ki = 8106 nM T20401 CCPO43 90654825 Ki > 50000 nM T20401 C4D2TM 90654826 Ki > 50000 nM T20401 C48XBN 90654827 Ki = 4870 nM T20401 CI8TG3 90654828 Ki > 50000 nM T20401 C6GFZ0 90654829 Ki = 87.3 nM T20401 C3Z1GS 90654830 Ki > 50000 nM T20401 C4JSW5 90655322 Ki = 336 nM T20401 C3QH0R 90655323 Ki = 296 nM T20401 CF0U7K 90655324 Ki = 274 nM T20401 C3OL7F 90656456 Ki = 38.5 nM T20401 CM10BY 90656457 Ki = 24 nM T20401 CGOV47 90656459 Ki = 10.3 nM T20401 CM3HC6 90656461 Ki = 79.7 nM T20401 CA9L3I 90656462 Ki = 130.5 nM T20401 C6F0AY 90656464 Ki = 11.2 nM T20401 CE0F5O 90656465 Ki = 8.6 nM T20401 CX4I7B 90656468 Ki = 51.5 nM T20401 CZ80KF 90656469 Ki = 158.4 nM T20401 CX4YM5 90656470 Ki = 32.4 nM T20401 CU31VY 90675933 Ki > 10000 nM T20401 C2XWG7 90675934 Ki > 10000 nM T20401 CH7R2B 90675935 Ki > 10000 nM T20401 CORQ94 90675936 Ki > 10000 nM T20401 CE39DC 90675937 Ki > 10000 nM T20401 CSU5K2 90675938 Ki > 10000 nM T20401 CE8S1J 90675939 Ki > 10000 nM T20401 C1H9FB 90675940 Ki > 10000 nM T20401 CPB36R 90675941 Ki > 10000 nM T20401 C3SJ1D 90677341 Ki = 7.1 nM T20401 CK1GA3 90677342 Ki = 11 nM T20401 C0CR6D 90681501 Ki = 730 nM T20401 C43EOS 90684366 Ki = 2300000 nM T20401 C7JD0F 91362447 Ki = 64000 nM T20401 C28FLQ 91498333 Ki > 10000 nM T20401 CE6LO5 91595667 Ki = 0.05 nM T20401 C3AYZ5 91811067 Ki = 2445 nM T20401 CQF98O 91827503 Ki = 6.8 nM T20401 C3I6NV 91827505 Ki = 7.7 nM T20401 CW1P4E 91827506 Ki = 4.7 nM T20401 CE2OY1 91995964 Ki = 86.2 nM T20401 CX45AP 92044053 Ki = 36 nM T20401 CEH68Q 93972064 Ki = 65.6 nM T20401 C28QRZ 101564149 Ki > 100000 nM T20401 CE8GH2 101874826 Ki = 6.5 nM T20401 C4W9FG 101874827 Ki = 5.3 nM T20401 CY7G8A 101874828 Ki = 3.7 nM T20401 C1TM8I 101874829 Ki = 4.2 nM T20401 CVZ3L5 101874830 Ki = 5.8 nM T20401 C2H5FC 101876957 Ki = 168 nM T20401 CDGZ03 101879106 Ki = 4.9 nM T20401 CY6ER7 101879108 Ki = 6.8 nM T20401 C04YZS 101913644 Ki = 65.3 nM T20401 CAC1W7 101913750 Ki > 50000 nM T20401 CQX8K1 101913751 Ki > 50000 nM T20401 CIP25Q 101913752 Ki > 50000 nM T20401 CTY15S 101913753 Ki > 50000 nM T20401 C49NEJ 101913754 Ki > 50000 nM T20401 CW5Q7L 101913755 Ki > 50000 nM T20401 CE90SD 102138248 Ki > 10000 nM T20401 CB1PK8 102151146 Ki = 13100 nM T20401 C0A6FY 102151151 Ki = 96100 nM T20401 CP1X9Y 102232756 Ki = 890 nM T20401 C1XV9H 102311866 Ki = 3200 nM T20401 CQBE51 102341119 Ki = 725 nM T20401 C2TX7A 102354117 Ki = 1.2 nM T20401 CK43QR 102405972 Ki = 541 nM T20401 C0CVO4 102480165 Ki > 100000 nM T20401 C6LUE5 109059506 Ki > 10000 nM T20401 CUY64D 109061586 Ki > 10000 nM T20401 CXN7Z8 110453853 Ki = 16.6 nM T20401 C6I0LD 112499923 Ki = 9.3 nM T20401 C8CFR6 112499924 Ki = 0.98 nM T20401 C74UZL 112684088 Ki = 0.1927 nM T20401 CK52CI 112686058 Ki = 0.4539 nM T20401 CP5B7N 112687648 Ki = 0.6722 nM T20401 CUR4V8 114816322 Ki > 10000 nM T20401 C3TZ9A 115950959 Ki = 2.2 nM T20401 CAO67C 118705769 Ki = 6.4 nM T20401 CW1D8A 118705770 Ki = 5.9 nM T20401 CTFB51 118705771 Ki = 5.5 nM T20401 C5NGT8 118705772 Ki = 5.3 nM T20401 C3G4ZN 118705773 Ki = 5.1 nM T20401 CBVD13 118705774 Ki = 7.2 nM T20401 C3KCZ6 118705775 Ki = 358 nM T20401 C5Z4QF 118705776 Ki = 479 nM T20401 CV4YN0 118705777 Ki = 75.9 nM T20401 C0IBQ8 118705778 Ki = 204 nM T20401 CH7LV5 118705779 Ki = 103 nM T20401 CU5SI9 118705780 Ki = 113 nM T20401 C6IGP0 118705781 Ki = 135 nM T20401 C7ZE2H 118705782 Ki = 64.1 nM T20401 C47QFN 118705783 Ki = 340 nM T20401 CO1P3T 118705784 Ki = 285 nM T20401 CK8E5C 118705785 Ki = 146 nM T20401 CS9G2U 118705786 Ki = 113 nM T20401 C1XV9M 118705787 Ki = 50 nM T20401 C7GW3Q 118705788 Ki = 53 nM T20401 CUIS94 118706141 Ki = 8.9 nM T20401 CET19U 118706142 Ki = 9.5 nM T20401 C6FBG3 118706893 Ki > 10000 nM T20401 C1CLV5 118706959 Ki > 10000 nM T20401 CLA5I2 118706960 Ki > 10000 nM T20401 C8GD4Y 118706961 Ki > 10000 nM T20401 CB0E4N 118706962 Ki > 10000 nM T20401 CFX37I 118707439 Ki = 9.8 nM T20401 CURF40 118707440 Ki = 91.9 nM T20401 C2SPI1 118707441 Ki = 83.5 nM T20401 CK7VG2 118707442 Ki = 197 nM T20401 CB6IF2 118707443 Ki = 83.1 nM T20401 C5O1TK 118707444 Ki = 71.3 nM T20401 C5VW3Z 118707445 Ki = 470 nM T20401 CM5Z7B 118707446 Ki = 847 nM T20401 CANH39 118707447 Ki = 71.2 nM T20401 CQO91H 118707448 Ki = 75.9 nM T20401 C2PU1D 118707449 Ki = 563 nM T20401 C8H7SM 118707452 Ki = 473 nM T20401 CYJ0I7 118707453 Ki = 384 nM T20401 C0R9FG 118707454 Ki = 452 nM T20401 CJI04D 118707455 Ki = 824 nM T20401 CO8AF6 118707456 Ki = 44 nM T20401 CJP1W6 118707457 Ki = 5100 nM T20401 C3G0AY 118707458 Ki = 5.9 nM T20401 CM1B4X 118707459 Ki = 29.4 nM T20401 C0WO2M 118707460 Ki = 4.4 nM T20401 CKV43U 118710106 Ki = 76.1 nM T20401 CBAQ59 118710108 Ki = 46.7 nM T20401 CPI7L3 118710135 Ki > 20000 nM T20401 C05ZCN 118710136 Ki > 20000 nM T20401 C45XHE 118710137 Ki > 20000 nM T20401 C84YKV 118710138 Ki > 20000 nM T20401 CFA76H 118710139 Ki = 2175 nM T20401 C0UWK2 118710140 Ki > 20000 nM T20401 CGJ59E 118710141 Ki > 20000 nM T20401 C64BUR 118710142 Ki > 20000 nM T20401 C1W2DB 118710143 Ki > 20000 nM T20401 CZ4F3O 118710144 Ki > 20000 nM T20401 CWR82N 118710145 Ki > 20000 nM T20401 C7R5FO 118710146 Ki > 20000 nM T20401 CD8U1O 118710147 Ki > 20000 nM T20401 C8YFH6 118710148 Ki > 20000 nM T20401 CLPC68 118710149 Ki > 20000 nM T20401 C8OH4V 118710150 Ki > 20000 nM T20401 C6CAQ4 118710151 Ki > 20000 nM T20401 CS0G7T 118710152 Ki > 20000 nM T20401 C3NPF1 118710200 Ki > 20000 nM T20401 C4YXF1 118710201 Ki > 20000 nM T20401 C1B5QL 118710202 Ki > 20000 nM T20401 CUJ42P 118710203 Ki = 25.5 nM T20401 CK23DF 118710598 Ki = 4.3 nM T20401 CS9MC2 118710599 Ki = 14.4 nM T20401 CW2D4O 118710600 Ki = 3.5 nM T20401 CTMF04 118710601 Ki = 3.9 nM T20401 CU2C9L 118710602 Ki = 6.1 nM T20401 CFCG50 118710603 Ki = 6 nM T20401 C2G5DI 118710604 Ki = 71.8 nM T20401 CY2S9V 118710605 Ki = 3.8 nM T20401 C5L6IK 118710606 Ki = 3.6 nM T20401 C6ZGB2 118711612 Ki = 50.4 nM T20401 CNS6L8 118711613 Ki = 755 nM T20401 CY0E8G 118711614 Ki = 142 nM T20401 CI71PW 118711615 Ki = 74.8 nM T20401 C1X7RI 118711616 Ki = 66.1 nM T20401 C7P6GM 118711617 Ki = 329 nM T20401 CYNA84 118711618 Ki = 32.7 nM T20401 CL38UN 118711619 Ki = 165 nM T20401 CGUV98 118711620 Ki = 30.1 nM T20401 CJ2UH6 118711621 Ki = 648 nM T20401 CH2RE7 118711622 Ki = 98.1 nM T20401 C1RWN4 118711623 Ki = 56.8 nM T20401 CR0I6S 118711624 Ki = 46.9 nM T20401 C8LQI3 118711625 Ki = 123 nM T20401 C5SEJ6 118711626 Ki = 26.9 nM T20401 C5TYE7 118711627 Ki = 142 nM T20401 C31WHN 118711637 Ki > 10000000 nM T20401 C7ZOH6 118712658 Ki = 421 nM T20401 C19IXJ 118712659 Ki = 413 nM T20401 CD5MB4 118712660 Ki = 629 nM T20401 C0EPI8 118712661 Ki = 552 nM T20401 CUO2I5 118714986 Ki = 1.3 nM T20401 CHL5P7 118714987 Ki = 1.8 nM T20401 CKGY64 118714988 Ki = 1.7 nM T20401 CQ3L5G 118714989 Ki = 208.4 nM T20401 CK9FR8 118714990 Ki = 233.8 nM T20401 CVM9K5 118714991 Ki = 208.9 nM T20401 CXP7N8 118714992 Ki = 12.1 nM T20401 C0OE2J 118714993 Ki = 122.9 nM T20401 CN26WF 118715053 Ki = 67.5 nM T20401 C6RIG2 118715054 Ki = 78.26 nM T20401 C9T4CK 118715055 Ki = 114.2 nM T20401 C19IQV 118715056 Ki = 96 nM T20401 CZ18GD 118716360 Ki = 94 nM T20401 CX6F4B 118716361 Ki = 525 nM T20401 CO4K8Z 118716362 Ki = 10 nM T20401 CR8HX4 118716363 Ki = 265 nM T20401 CYH2P1 118716364 Ki = 110 nM T20401 C61BOY 118716365 Ki = 190 nM T20401 C8PJC3 118716366 Ki = 5 nM T20401 C9HP7J 118716367 Ki = 6400 nM T20401 CTS52R 118716368 Ki = 20000 nM T20401 CHI60Z 118716369 Ki = 185 nM T20401 CA1UY4 118716496 Ki = 8.3 nM T20401 CVR32C 118716497 Ki = 8.9 nM T20401 CT1RQ6 118716498 Ki = 41.8 nM T20401 CG10AC 118716499 Ki = 17.2 nM T20401 CV89MK 118716500 Ki = 9.4 nM T20401 C57YMW 118716501 Ki = 150 nM T20401 CQ73KL 118716502 Ki = 8.5 nM T20401 CXE59K 118716504 Ki = 589 nM T20401 CONM87 118716505 Ki = 192 nM T20401 CQ3I7N 118716509 Ki = 5.8 nM T20401 C72KER 118716510 Ki = 4.5 nM T20401 C0RJI1 118716511 Ki = 5.2 nM T20401 CFU0Z8 118716512 Ki = 4.5 nM T20401 CXU4D7 118716513 Ki = 9.3 nM T20401 C86KQZ 118716514 Ki > 10000 nM T20401 C9HLA8 118716891 Ki = 94 nM T20401 CJ0YC9 118716892 Ki = 86 nM T20401 CJ8TZ3 118716893 Ki > 10000 nM T20401 C0X1WQ 118716894 Ki > 10000 nM T20401 CDG4L8 118716895 Ki = 94 nM T20401 CFD26B 118716950 Ki = 682 nM T20401 C20YBM 118716951 Ki = 664 nM T20401 C0V1ZT 118716952 Ki = 710 nM T20401 CH9BW0 118716953 Ki = 63.5 nM T20401 CXB89Y 118716954 Ki = 498 nM T20401 C8CKU2 118716955 Ki = 701 nM T20401 CYN29C 118716960 Ki = 403 nM T20401 C4AC7H 118716961 Ki = 709 nM T20401 CJ9O3I 118716962 Ki = 713 nM T20401 C6RJ9W 118716964 Ki = 652 nM T20401 CMVW90 118716999 Ki = 91 nM T20401 CBKN39 118717000 Ki > 10000 nM T20401 C6N8CF 118717001 Ki > 10000 nM T20401 CL3P7I 118717002 Ki = 85 nM T20401 C2H0NP 118717003 Ki > 10000 nM T20401 CXRD23 118719969 Ki = 33.9 nM T20401 C4Z6DI 118719970 Ki = 37.6 nM T20401 C2HJ4Y 118719971 Ki > 10000 nM T20401 CD1OH8 118719972 Ki > 10000 nM T20401 C0R8JN 118719973 Ki = 7380 nM T20401 CMR0H2 118719974 Ki = 8160 nM T20401 CI3QG5 118719975 Ki > 10000 nM T20401 C06YTV 118719976 Ki > 10000 nM T20401 C25BJT 118721385 Ki = 10.9 nM T20401 CI4W0E 118721386 Ki = 31.5 nM T20401 CFRX59 118721387 Ki = 39.9 nM T20401 C5SYD7 118721388 Ki = 10.4 nM T20401 CNT18B 118721389 Ki = 142 nM T20401 CYC50E 118721390 Ki = 3.8 nM T20401 CYL0W1 118721391 Ki = 2.3 nM T20401 C1HN6R 118721392 Ki = 2.3 nM T20401 C2WLI4 118721393 Ki = 2.7 nM T20401 CQVS30 118721394 Ki = 2.5 nM T20401 CL2Q8M 118721395 Ki = 7.3 nM T20401 CAG5L6 118721396 Ki = 9.3 nM T20401 CJ63BR 118721397 Ki = 139 nM T20401 C14ZNT 118721398 Ki = 48.1 nM T20401 C1J6IX 118721399 Ki = 4736 nM T20401 CVJ92D 118721400 Ki = 27 nM T20401 C5F7PT 118721401 Ki = 4821 nM T20401 C5AFR3 118721402 Ki = 1386 nM T20401 C29EYL 118721403 Ki = 64 nM T20401 C8GYO9 118721404 Ki = 13.7 nM T20401 CSZ7Q0 118721405 Ki = 15.8 nM T20401 CY3ZW6 118721406 Ki = 8.5 nM T20401 C4T9IR 118721407 Ki = 85.1 nM T20401 CNPB81 118721408 Ki = 11.6 nM T20401 CP40JF 118722001 Ki > 10000 nM T20401 CXTR97 118723294 Ki = 5 nM T20401 C42JBV 118723295 Ki = 5.1 nM T20401 CVDC56 118723296 Ki = 5.5 nM T20401 C2RG7F 118723303 Ki = 5 nM T20401 C0CMO4 118723304 Ki = 4.6 nM T20401 CC7RH0 118723305 Ki = 3.9 nM T20401 CU0R8X 118723306 Ki = 215 nM T20401 C67LPC 118723308 Ki = 43.3 nM T20401 C0D1SQ 118724328 Ki = 6 nM T20401 C89YTC 118724329 Ki = 6.1 nM T20401 CBT87C 118724330 Ki = 41 nM T20401 C49AWZ 118724331 Ki = 6.9 nM T20401 CP9X5K 118728047 Ki = 35.8 nM T20401 CUA3S7 118728048 Ki = 41.7 nM T20401 C2K3DO 118728049 Ki = 24.3 nM T20401 CZTN86 118728050 Ki = 17.3 nM T20401 C0CUV2 118728051 Ki = 48.7 nM T20401 CGU5O0 118728053 Ki = 18.9 nM T20401 CGQ69F 118728055 Ki = 65.9 nM T20401 C2JEW0 118728057 Ki = 80.1 nM T20401 CCBJ19 118728058 Ki = 45.4 nM T20401 CKJ8S9 118728060 Ki = 80.5 nM T20401 C0O3BI 118728062 Ki = 8.9 nM T20401 CH2E8F 118728064 Ki = 47.9 nM T20401 C4JM1O 118728066 Ki = 13.2 nM T20401 C67YPT 118728068 Ki = 60.2 nM T20401 CML9F8 118728070 Ki = 78.5 nM T20401 CA52IR 118728072 Ki = 67.2 nM T20401 CVE9H5 118728074 Ki = 48.1 nM T20401 CS9ZW3 118728500 Ki > 10000 nM T20401 CI7MY8 118728501 Ki > 10000 nM T20401 CZE9K8 118728502 Ki > 10000 nM T20401 C8S9JV 118728503 Ki = 422 nM T20401 COJB53 118728998 IC50 = 121.5 nM T20401 C4GJ2A 118728999 IC50 = 110.2 nM T20401 C16CPW 118729000 Ki = 90.3 nM T20401 CRH8X5 118729001 IC50 = 130.6 nM T20401 CD97RL 118729002 Ki = 48.09 nM T20401 C19HNU 118729003 IC50 = 126.5 nM T20401 C8IJ7W 118729004 IC50 = 110.9 nM T20401 CZLP09 118729005 Ki = 138 nM T20401 C1W9DT 118729006 Ki = 122.4 nM T20401 CS30QV 118729007 Ki = 58.3 nM T20401 C40AIB 118729374 Ki > 10000 nM T20401 CO3Z5E 118729375 Ki > 10000 nM T20401 C6S0DR 118729376 Ki > 10000 nM T20401 CVXO79 118729377 Ki > 10000 nM T20401 C62BGK 118729378 Ki > 10000 nM T20401 C4D9EP 118729379 Ki > 10000 nM T20401 C2TOH7 118729380 Ki > 10000 nM T20401 C5P9ND 118729381 Ki > 10000 nM T20401 C2XLV4 118729382 Ki > 10000 nM T20401 CVLK60 118729383 Ki > 10000 nM T20401 C8U7SE 118729384 Ki > 10000 nM T20401 CV7OS1 118729385 Ki > 10000 nM T20401 C7Z2OR 118729386 Ki > 10000 nM T20401 CHE1K4 118729473 Ki = 26 nM T20401 C9V8MA 118729474 Ki = 41.6 nM T20401 C8GJP5 118729475 Ki = 22.1 nM T20401 C4MEZ0 118729476 Ki = 52.1 nM T20401 CE3IV5 118729477 Ki = 1785 nM T20401 C5DM9L 118731312 Ki = 0.2 nM T20401 C7EX8M 118732578 Ki = 83 nM T20401 C0A2SM 118732579 Ki = 201 nM T20401 CV2JZ8 118732580 Ki = 114 nM T20401 C2GNO4 118732581 Ki = 201 nM T20401 CES83M 118732582 Ki = 9.1 nM T20401 CF2WQ4 118732583 Ki = 2.7 nM T20401 CEN7K8 118733205 IC50 = 82 nM T20401 C08EZC 118733945 Ki > 10000 nM T20401 C3F1DU 118733947 Ki > 10000 nM T20401 C4OL1A 118733948 Ki > 10000 nM T20401 CP25HS 118733949 Ki > 10000 nM T20401 CY3H4E 118736318 Ki = 600 nM T20401 C8HY4S 118736320 Ki = 433 nM T20401 C7F5JH 118736322 Ki = 819 nM T20401 C7MDJ3 118736324 Ki = 315 nM T20401 CQM67J 118736325 Ki = 8.5 nM T20401 CKY90W 118736326 Ki = 7.6 nM T20401 CY4B1U 118736327 Ki = 6.6 nM T20401 CRZ1T6 118736328 Ki = 29.5 nM T20401 CFDB97 118737265 Ki > 10000 nM T20401 CVGF86 118737267 Ki > 10000 nM T20401 C6B8WR 118737268 Ki > 10000 nM T20401 CWEM68 118737269 Ki > 10000 nM T20401 C6PXT8 118737270 Ki > 10000 nM T20401 CWP7Q1 118737271 Ki > 10000 nM T20401 CAB65M 118737272 Ki > 10000 nM T20401 CHR0I7 118737273 Ki > 10000 nM T20401 C72BLG 118737274 Ki > 10000 nM T20401 C4TD0Q 118737275 Ki > 10000 nM T20401 CZ1J0U 118737276 Ki > 10000 nM T20401 CHN09Y 118737277 Ki > 10000 nM T20401 CMR62B 118737278 Ki > 10000 nM T20401 C1CV3E 118737279 Ki > 10000 nM T20401 CUQ7H9 119082247 Ki = 7.9 nM T20401 CP8Y5U 119090745 Ki > 10000 nM T20401 C4K6CG 119943184 Ki > 10000 nM T20401 CHX4Y2 121382833 Ki > 50000 nM T20401 CNEJ87 121382878 Ki = 9 nM T20401 CBHM75 121382881 Ki = 450 nM T20401 C13GKC 121382882 Ki = 553 nM T20401 C8QTR4 121382883 Ki = 747 nM T20401 C96ANJ 121382897 Ki > 50000 nM T20401 CUS64J 121382999 Ki = 90.5 nM T20401 C6C4WE 121383002 Ki = 15.7 nM T20401 CG48HD 122164592 Ki = 780 nM T20401 C86KHO 122179484 Ki = 3.9 nM T20401 C0OX5C 122179485 Ki = 0.77 nM T20401 CK92MV 122179845 Ki > 50000 nM T20401 C10UQY 122179846 Ki = 7070 nM T20401 CLV96C 122179847 Ki > 50000 nM T20401 C2RT1Y 122179848 Ki > 50000 nM T20401 C06ZSC 122179849 Ki > 50000 nM T20401 C74RAE 122179850 Ki > 50000 nM T20401 C6NM0Q 122179851 Ki > 50000 nM T20401 CYP3B0 122179852 Ki > 50000 nM T20401 CMP05I 122179853 Ki > 50000 nM T20401 C2TGN6 122179854 Ki > 50000 nM T20401 CAH3I1 122179855 Ki > 50000 nM T20401 CPKX90 122179856 Ki = 0.0603 nM T20401 CQ2P5O 122179857 Ki = 0.1561 nM T20401 CVB9C4 122179858 Ki = 0.0888 nM T20401 CO6QP7 122179859 Ki = 0.0488 nM T20401 CP01MN 122179860 Ki = 0.1051 nM T20401 CJG71H 122179861 Ki = 0.1368 nM T20401 C8YJ9B 122180166 Ki > 10000 nM T20401 CHON20 122180167 Ki > 10000 nM T20401 C9L2TG 122180168 Ki > 10000 nM T20401 C9L3OY 122180169 Ki > 10000 nM T20401 CJ1X2F 122180170 Ki > 10000 nM T20401 CVCX92 122180171 Ki > 10000 nM T20401 C6LEA3 122180172 Ki > 10000 nM T20401 CV8Z4I 122182643 Ki = 226 nM T20401 CV96QP 122182644 Ki = 9.2 nM T20401 CA91HP 122182645 Ki = 9.3 nM T20401 C08EBQ 122182646 Ki = 9 nM T20401 CSJA24 122182647 Ki = 45.4 nM T20401 CDM51W 122182648 Ki = 8.9 nM T20401 C3E9FK 122182649 Ki = 8.6 nM T20401 CUF5N9 122182650 Ki = 4.7 nM T20401 C5BRH0 122182651 Ki = 8.6 nM T20401 C45DQE 122182654 Ki = 4.1 nM T20401 CDRF43 122182655 Ki = 4.7 nM T20401 CQ83BJ 122182656 Ki = 3.5 nM T20401 CH4Z8B 122182657 Ki = 3.7 nM T20401 CU71LK 122182658 Ki = 3.5 nM T20401 CY1NK4 122182659 Ki = 4.7 nM T20401 CP4I8D 122184891 Ki = 10.9 nM T20401 CZ2RM0 122184892 Ki = 0.6 nM T20401 CFQ4R3 122184893 Ki = 1.5 nM T20401 C69UQF 122184894 Ki = 1.4 nM T20401 CNF20A 122184895 Ki = 3.1 nM T20401 CJAL95 122184896 Ki = 5.5 nM T20401 C51LFX 122184933 Ki = 0.17 nM T20401 CTQP23 122184934 Ki = 0.54 nM T20401 CL49QM 122184935 Ki = 1.1 nM T20401 CVN28C 122184936 Ki = 1.7 nM T20401 CU4S6Y 122184937 Ki = 0.26 nM T20401 C4VWG9 122184938 Ki = 0.3 nM T20401 C7H8ZI 122184984 Ki = 11.7 nM T20401 CX76HF 122184985 Ki = 71.9 nM T20401 C1KOF6 122184986 Ki = 18.2 nM T20401 C01CWK 122184987 Ki = 16.9 nM T20401 CVTY87 122184988 Ki = 15.9 nM T20401 CM5A7F 122184989 Ki = 11.1 nM T20401 CYM65N 122184990 Ki = 11.2 nM T20401 CQ9YU1 122184991 Ki = 9.1 nM T20401 C83GXC 122184992 Ki = 1.2 nM T20401 CTV40W 122184993 Ki = 1.1 nM T20401 CWM21G 122184994 Ki = 1 nM T20401 C19LDQ 122184995 Ki = 81.6 nM T20401 C7UE2C 122184996 Ki = 5935.6 nM T20401 CWBN52 122184997 Ki = 519.5 nM T20401 C1CI4W 122184998 Ki = 1427.7 nM T20401 CWJ94V 122185033 Ki = 10 nM T20401 C3G8EB 122185233 Ki = 778500 nM T20401 C9PG8Z 122185234 Ki = 2146 nM T20401 C93KBM 122185235 Ki = 91.5 nM T20401 CX6Z5Y 122185236 Ki = 15.4 nM T20401 CFPV38 122185237 Ki = 14.9 nM T20401 CVZ70D 122185238 Ki = 71.8 nM T20401 C14OHP 122185239 Ki = 14.4 nM T20401 CB63WU 122185240 Ki = 10.7 nM T20401 CE3Q1J 122185241 Ki = 51.8 nM T20401 CNG63S 122185242 Ki = 15.5 nM T20401 CY7H0T 122185243 Ki = 14.4 nM T20401 C2ME1I 122185244 Ki = 37.5 nM T20401 C0EPT7 122185245 Ki = 0.07 nM T20401 CI1AL4 122185246 Ki = 26.9 nM T20401 CM43CE 122185684 Ki > 10000 nM T20401 CSQ43L 122185685 Ki > 10000 nM T20401 CCA9I1 122185686 Ki > 10000 nM T20401 CLIR24 122185687 Ki = 942 nM T20401 C5NWU9 122185688 Ki = 788 nM T20401 CY70TU 122185689 Ki = 98 nM T20401 CD94UC 122185690 Ki = 707 nM T20401 C8TIP4 122185692 Ki = 507 nM T20401 CE7W6O 122185694 Ki = 9338 nM T20401 CV2G7S 122185695 Ki = 958 nM T20401 C1M5JR 122185696 Ki = 16 nM T20401 CMB32C 122185697 Ki > 10000 nM T20401 C1FR9Q 122185698 Ki > 10000 nM T20401 CY2D9L 122185699 Ki > 10000 nM T20401 C2NUJ9 122185700 Ki > 10000 nM T20401 C6VE0K 122185734 IC50 = 514 nM T20401 C9AVI2 122185735 IC50 = 403 nM T20401 CHBC74 122185771 Ki = 13 nM T20401 CZM98F 122185772 Ki > 10000 nM T20401 CP8Y5E 122185773 Ki > 10000 nM T20401 CK2Q7M 122185774 Ki > 10000 nM T20401 CF4L0N 122185776 Ki > 10000 nM T20401 C7T4BF 122185778 Ki > 10000 nM T20401 C4TZ6G 122185779 Ki > 10000 nM T20401 CUI73A 122187162 Ki = 0.01 nM T20401 C1Q7AX 122187163 Ki = 0.02 nM T20401 CO6P7A 122187164 Ki = 0.009 nM T20401 C9LN8Q 122187165 Ki = 0.008 nM T20401 COK6D7 122187166 Ki = 7.1 nM T20401 C7NV8G 122187167 Ki = 63.9 nM T20401 C6XKH1 122187168 Ki = 283 nM T20401 C5KMW2 122187169 Ki = 4420 nM T20401 CSA78D 122187170 Ki = 8860 nM T20401 C5V7SZ 122187171 Ki = 58.2 nM T20401 C6FMG1 122187172 Ki = 0.01 nM T20401 CVG1U0 122187173 Ki = 0.28 nM T20401 CR8NT0 122187174 Ki = 0.01 nM T20401 CWSM36 122187175 Ki = 0.05 nM T20401 CT59AR 122187176 Ki = 6.3 nM T20401 C93ESN 122187177 Ki = 4.8 nM T20401 CL0JF6 122187178 Ki = 0.01 nM T20401 CQ81UP 122187179 Ki = 0.01 nM T20401 CIE0W8 122187180 Ki = 0.02 nM T20401 CNSU27 122187181 Ki = 0.01 nM T20401 C7LDH1 122187182 Ki = 2.5 nM T20401 CG9T3N 122187183 Ki = 0.01 nM T20401 CBE9U8 122187184 Ki = 0.02 nM T20401 C13USE 122187185 Ki = 0.03 nM T20401 CE36PK 122187423 Ki = 88.1 nM T20401 CDS2I6 122187424 Ki = 14.7 nM T20401 CMF63L 122187425 Ki = 721 nM T20401 C7Q9TP 122187426 Ki = 5.4 nM T20401 C04HSI 122187596 Ki = 5 nM T20401 CZ74KO 122187597 Ki = 1 nM T20401 C07OYV 122187598 Ki = 3 nM T20401 CO6AT2 122187599 Ki = 5 nM T20401 C7WJ4B 122187600 Ki = 6 nM T20401 CZ0Y1G 122187601 Ki = 4 nM T20401 CWF7Z0 122187602 Ki = 5 nM T20401 C07ZNW 122187603 Ki = 8 nM T20401 C7K6TV 122187604 Ki = 217 nM T20401 CX69YT 122187605 Ki = 3 nM T20401 C8XN0F 122187606 Ki = 6 nM T20401 CVT13C 122187607 Ki = 4 nM T20401 CB2DT8 122187638 Ki = 1.7 nM T20401 C0G4CQ 122187639 Ki = 136 nM T20401 CQSV13 122187640 Ki = 0.75 nM T20401 CH74EW 122187641 Ki = 4.1 nM T20401 CH3C8V 122187642 Ki = 6.8 nM T20401 CP01NQ 122187643 Ki = 5.7 nM T20401 CRM3S4 122188878 Ki = 3.7 nM T20401 C5UF1Q 122188879 Ki = 6.3 nM T20401 CQB9A8 122188880 Ki = 74.8 nM T20401 C1SFD4 122188881 Ki = 1.8 nM T20401 CIE7L0 122188882 Ki = 52.3 nM T20401 C6MPI4 122189078 Ki > 40000 nM T20401 C9V7WT 122189088 Ki > 40000 nM T20401 C1QZV7 122189098 Ki > 40000 nM T20401 CN16RY 122189300 Ki = 11.2 nM T20401 CYN3T8 122189301 Ki = 5.89 nM T20401 CSW9D1 122189302 Ki = 9.5 nM T20401 C6USQ7 122189303 Ki = 10.4 nM T20401 CQ4X1G 122189304 Ki = 15.1 nM T20401 C5XT3S 122192640 Ki = 640 nM T20401 C1LCB9 122192641 Ki = 650 nM T20401 CP51XT 122192642 Ki = 500 nM T20401 C5GKT0 122192643 Ki = 100 nM T20401 C3RZM8 122192644 Ki = 960 nM T20401 CHLG86 122192645 Ki = 370 nM T20401 CTK4J8 122192646 Ki = 600 nM T20401 CVNQ49 122192647 Ki = 480 nM T20401 CX3A0N 122192648 Ki = 470 nM T20401 CU3F1V 122192649 Ki = 380 nM T20401 CQ4NT8 122192650 Ki = 390 nM T20401 C2REU8 122192651 Ki = 250 nM T20401 CL5P4T 122192652 Ki = 450 nM T20401 C0KF5I 122192653 Ki = 430 nM T20401 CT64DB 122192654 Ki = 500 nM T20401 CX05RY 122192671 Ki > 10000 nM T20401 CE9ZC4 122192672 Ki > 10000 nM T20401 CUW2B9 122192673 Ki > 10000 nM T20401 CKU76Q 122192674 Ki > 10000 nM T20401 C49KGU 122192675 Ki > 10000 nM T20401 CB0J2T 122192676 Ki > 10000 nM T20401 CS63LF 122192677 Ki > 10000 nM T20401 C4T3IO 122192678 Ki = 99.6 nM T20401 CTZ4L6 122192679 Ki > 10000 nM T20401 C62VGD 122192680 Ki > 10000 nM T20401 CYND20 122192681 Ki > 10000 nM T20401 CLV5O9 122192682 Ki = 9743 nM T20401 CH1N0C 122193189 Ki > 50000 nM T20401 C19HVL 122193190 Ki > 50000 nM T20401 C5TQJ1 122193251 Ki > 50000 nM T20401 C8XCL0 122193252 Ki > 50000 nM T20401 CH4IV8 122194771 Ki = 9 nM T20401 CQ7N0L 122194772 Ki = 42 nM T20401 CI5K2F 122194773 Ki = 5.3 nM T20401 CV51IU 122194774 Ki = 11.5 nM T20401 C7OFR6 122194775 Ki = 4.3 nM T20401 C81HNW 122194776 Ki = 4.9 nM T20401 C8J5QV 122194777 Ki = 454 nM T20401 CV1C9T 122194778 Ki = 7.8 nM T20401 CJC1W3 122194779 Ki = 6.6 nM T20401 CU1TV5 122194780 Ki = 50.6 nM T20401 C4C1BE 122194781 Ki = 814 nM T20401 CR9I5Q 122194782 Ki = 6.9 nM T20401 C8SVY4 122194783 Ki = 63.3 nM T20401 C7HT8B 122194784 Ki = 5.9 nM T20401 CW8P3R 122194785 Ki = 39.7 nM T20401 COAK34 122194786 Ki = 5.2 nM T20401 CPN73S 122199224 Ki = 1025 nM T20401 CC1UO6 122226187 Ki = 910 nM T20401 C7T0FH 122226188 Ki = 17700 nM T20401 C3EG2B 122226189 Ki = 19100 nM T20401 C18KAD 122367673 Ki = 6.43 nM T20401 CPN5F4 122367675 Ki = 8.91 nM T20401 C26IUP 122386532 Ki > 100000 nM T20401 CGE1Q6 122707121 Ki = 2.1 nM T20401 C1JBF7 122707123 Ki = 2.5 nM T20401 CGPI62 123372490 Ki = 1 nM T20401 CPO7N5 124125214 IC50 > 10000 nM T20401 CV4GW7 126961712 Ki = 3.3 nM T20401 C0FD4E 126961713 Ki = 3.6 nM T20401 CD3HF0 127024855 Ki = 2.85 nM T20401 CXY79J 127024883 Ki > 10000 nM T20401 CK9C7T 127024884 Ki > 10000 nM T20401 C50MSQ 127024885 Ki > 10000 nM T20401 C4N6WJ 127024886 Ki = 1749 nM T20401 C5AES0 127024887 Ki > 10000 nM T20401 CHU95V 127024991 Ki = 764 nM T20401 CP8O7D 127024992 Ki = 324 nM T20401 CRHW31 127024993 Ki = 0.95 nM T20401 C57BLH 127025130 Ki = 7.4 nM T20401 C0T4VY 127025177 Ki = 3.26 nM T20401 CRTB63 127025292 Ki = 14.2 nM T20401 CAO31Y 127025293 Ki = 11.1 nM T20401 CL0ZR4 127025295 Ki = 18 nM T20401 C9JNZ5 127025296 Ki = 0.68 nM T20401 C04USY 127025300 Ki = 5.9 nM T20401 CDB1Z9 127025301 Ki = 0.25 nM T20401 CYK6H1 127025302 Ki = 10.8 nM T20401 C7UF0B 127025480 Ki > 10000 nM T20401 CY7DI6 127025481 Ki = 1.15 nM T20401 C6M4SW 127025591 Ki = 10.4 nM T20401 CUPA95 127025592 Ki = 9.4 nM T20401 CWP36V 127025593 Ki = 0.61 nM T20401 C0DL8N 127026696 Ki = 2.15 nM T20401 C95QVS 127026977 Ki = 5390 nM T20401 C09PAM 127026978 Ki = 4220 nM T20401 CS96JF 127026979 Ki > 50000 nM T20401 CRB80M 127026980 Ki = 638 nM T20401 C0RBK5 127027010 Ki = 140 nM T20401 C0WY9H 127027097 Ki = 2.1 nM T20401 CP84DU 127027288 Ki = 7450 nM T20401 CH30BV 127027289 Ki = 96 nM T20401 CM72RV 127027290 Ki = 63.2 nM T20401 CO3IJ7 127027291 Ki = 218 nM T20401 CTS74J 127027656 Ki = 1.86 nM T20401 CL9G1Y 127027664 Ki = 0.98 nM T20401 C9G5HM 127027733 Ki = 2.16 nM T20401 CT0E5I 127027734 Ki = 1.91 nM T20401 C2C3GA 127027735 Ki = 2.9 nM T20401 CT1Q7O 127027978 Ki = 5.19 nM T20401 CRL3B5 127028045 Ki = 2.89 nM T20401 C4O2XT 127028951 Ki > 10000 nM T20401 CFIW54 127029020 Ki = 10.2 nM T20401 C5RBS3 127029021 Ki = 764 nM T20401 CPA6G5 127029022 Ki = 0.7 nM T20401 C74ZGJ 127029023 Ki = 0.84 nM T20401 CN3PH9 127029250 Ki > 10000 nM T20401 CTY1H9 127029498 Ki = 9.4 nM T20401 CC1E7F 127029514 Ki = 2.56 nM T20401 C1J0RU 127029568 Ki = 0.35 nM T20401 CE38AJ 127030670 Ki = 2.8 nM T20401 CKL6D3 127030963 Ki = 462 nM T20401 CWFJ07 127030973 Ki = 514 nM T20401 C4T2KL 127031264 Ki = 2.69 nM T20401 C8G3YC 127031289 Ki = 101 nM T20401 CHG8P6 127031292 Ki = 491 nM T20401 C8SA4R 127031846 Ki = 2.19 nM T20401 C2ILH1 127031859 Ki = 1.82 nM T20401 C4PZ0V 127032697 Ki = 432 nM T20401 CNH03L 127033707 Ki = 2.43 nM T20401 C8CN4T 127033708 Ki = 2.33 nM T20401 C1C8XD 127034555 Ki = 1.88 nM T20401 CC4J3A 127034556 Ki = 1.64 nM T20401 CO48QN 127034557 Ki = 2.04 nM T20401 CRN4X6 127034558 Ki = 1.92 nM T20401 CTAR42 127034559 Ki = 2.66 nM T20401 C67ZWL 127034560 Ki = 2.79 nM T20401 CS2K4U 127034999 Ki > 10000 nM T20401 CFG39M 127035855 Ki = 4957 nM T20401 C6MH2V 127035856 Ki = 8884 nM T20401 CVO4B6 127035857 Ki > 10000 nM T20401 CQC6P9 127035858 Ki > 10000 nM T20401 C7YA3N 127035859 Ki = 7681 nM T20401 CXZI89 127035860 Ki > 10000 nM T20401 C5KLP8 127035861 Ki = 8528 nM T20401 CTVN28 127036466 Ki = 8 nM T20401 CWPY69 127036947 Ki = 8.5 nM T20401 CL76JS 127037630 Ki > 10000 nM T20401 CY1JU3 127037755 Ki = 28.3 nM T20401 C0UQ7W 127037756 Ki > 10000 nM T20401 CQUE67 127037757 Ki > 10000 nM T20401 CL3Q0T 127037870 Ki = 397 nM T20401 CK3VW1 127037881 Ki = 11.7 nM T20401 CN36JQ 127037910 IC50 > 10000 nM T20401 CTSR32 127038212 Ki = 6.8 nM T20401 CQTS23 127038553 Ki = 19.1 nM T20401 COVZ04 127038617 IC50 = 4600 nM T20401 CG8B3V 127039153 Ki = 8.9 nM T20401 CIO74C 127039154 Ki = 10.5 nM T20401 C0L8NH 127039155 Ki = 13.8 nM T20401 CJ2UY6 127039306 IC50 = 2200 nM T20401 CS96GU 127039479 Ki > 10000 nM T20401 C6WCG5 127039856 Ki = 7.7 nM T20401 C4NQ5H 127039905 Ki = 1.3 nM T20401 C3J8ET 127040041 Ki > 10000 nM T20401 C0P5HB 127040227 Ki = 0.31 nM T20401 CCD87Q 127040239 Ki = 7.7 nM T20401 C97DAS 127040240 Ki = 7.5 nM T20401 C9OZP8 127040553 Ki = 5.2 nM T20401 C4SH5D 127040554 Ki = 6.9 nM T20401 CCO9S8 127040555 Ki = 5.8 nM T20401 CB8TU5 127040913 IC50 = 700 nM T20401 CY9D7F 127040981 IC50 = 3800 nM T20401 CJR5F2 127040982 IC50 = 10000 nM T20401 C12SMV 127041490 Ki = 0.69 nM T20401 CUL2T4 127041605 IC50 = 700 nM T20401 CSJ3V0 127041732 Ki = 127 nM T20401 CG75VH 127041733 Ki = 88 nM T20401 CQC6A4 127042329 Ki > 10000 nM T20401 CZ6F5V 127042845 IC50 = 500 nM T20401 CRZK01 127043469 Ki = 9.1 nM T20401 C41YOV 127044252 Ki = 2.7 nM T20401 CMTC13 127044428 Ki = 4.2 nM T20401 C7KU0Z 127044429 Ki = 1.5 nM T20401 CJO3U8 127044444 Ki = 2.5 nM T20401 CAXM67 127044445 Ki = 1.9 nM T20401 CHP23N 127044446 Ki > 40000 nM T20401 C1T4LU 127044499 Ki = 10.7 nM T20401 CI3PD8 127044664 Ki = 1.2 nM T20401 CU5B2G 127044665 Ki = 0.86 nM T20401 CM9QJ3 127044834 Ki = 1 nM T20401 C5HIY4 127044835 Ki = 0.69 nM T20401 CKW0B5 127044836 Ki = 31.9 nM T20401 C0KQB1 127044932 Ki = 0.58 nM T20401 C4WZJ7 127044997 Ki = 0.78 nM T20401 C1LIQ5 127044998 Ki = 0.91 nM T20401 C3S2GY 127044999 Ki = 0.71 nM T20401 C62OLS 127045037 Ki = 0.47 nM T20401 C31FCL 127045083 Ki = 288 nM T20401 CT9KP2 127045237 Ki = 0.41 nM T20401 C17GLC 127045238 Ki = 0.62 nM T20401 C1U0VA 127045339 Ki = 2.3 nM T20401 C5EX6R 127048632 Ki = 16.8 nM T20401 CG10PI 127048878 Ki = 106.06 nM T20401 C3PHY8 127048879 Ki = 153.71 nM T20401 COLX43 127048880 Ki = 18.93 nM T20401 CBJ74P 127048881 Ki = 48.79 nM T20401 CK1X5H 127048994 Ki = 4.3 nM T20401 C2XK0I 127048995 Ki = 2.8 nM T20401 CY4P2X 127048996 Ki = 0.8 nM T20401 C6JB5S 127048997 Ki = 3.4 nM T20401 C1XE4W 127049197 Ki = 61.55 nM T20401 CCX35L 127049198 Ki = 1868.14 nM T20401 CRE6O9 127049213 Ki = 17.09 nM T20401 CP40EB 127049242 Ki = 12.9 nM T20401 CLFB54 127049248 Ki = 66.6 nM T20401 C1T3WG 127049310 Ki = 2.3 nM T20401 CKO03S 127049970 Ki = 55.4 nM T20401 CP8KG9 127049971 Ki = 2.4 nM T20401 CY5MI3 127049999 Ki > 50000 nM T20401 C5CNP8 127050174 Ki = 153.26 nM T20401 C9EJ6L 127050230 Ki = 9.9 nM T20401 CH07TV 127050456 Ki = 21.2 nM T20401 CP8U0D 127050457 Ki = 17.46 nM T20401 C65PAS 127050458 Ki = 18.45 nM T20401 C7MI5Q 127050568 Ki = 4.4 nM T20401 C1RGQ6 127050569 Ki = 8.7 nM T20401 CB5W0L 127050570 Ki = 0.5 nM T20401 CUG58A 127050571 Ki = 2.8 nM T20401 CJP49X 127050777 Ki = 15.66 nM T20401 CER02F 127050778 Ki = 95.64 nM T20401 CG17IO 127050812 Ki = 1764 nM T20401 C8X6CY 127050822 Ki = 9.3 nM T20401 C9FZ4E 127050900 Ki = 2.2 nM T20401 C4IA5N 127051119 Ki = 37.1 nM T20401 CRDQ30 127051120 Ki = 8.7 nM T20401 CJ0EQ7 127051501 Ki = 5110 nM T20401 CUWE95 127051804 Ki = 6.8 nM T20401 COBU26 127051805 Ki = 4.8 nM T20401 C7SIY6 127051806 Ki = 5.5 nM T20401 C5Y4DI 127051953 Ki = 8.6 nM T20401 CJ7WT3 127052106 Ki = 32.2 nM T20401 CM21NF 127052276 Ki = 1751.72 nM T20401 C90PLX 127052516 Ki > 50000 nM T20401 CFQ75A 127052517 Ki = 4520 nM T20401 C26TUM 127052712 Ki = 2.7 nM T20401 C7PS8D 127052713 Ki = 4.4 nM T20401 C32ART 127052714 Ki = 47.3 nM T20401 CEC30I 127052811 Ki > 50000 nM T20401 C5CW4K 127052812 Ki > 50000 nM T20401 C5V7QI 127052813 Ki = 1350 nM T20401 CI24ZM 127052900 Ki = 13.23 nM T20401 CEVZ36 127052901 Ki = 757.83 nM T20401 CX1Z2E 127052917 Ki = 16.89 nM T20401 CM8FI7 127052918 Ki = 19.04 nM T20401 CUOZ60 127052919 Ki = 17.49 nM T20401 C9D6CB 127053004 Ki = 5.1 nM T20401 CHN5K6 127567366 Ki = 1.8 nM T20401 C4JC3W 127573780 Ki = 51.4 nM T20401 C85FAK 129009671 Ki = 1 nM T20401 C7R6LY 129009672 Ki = 1.2 nM T20401 C2B6XM 129673327 Ki > 10000 nM T20401 CJC35Q 129856021 Ki > 10000 nM T20401 CCF61S 129883275 Ki = 92.5 nM T20401 CNB2M7 131839635 Ki = 5.5 nM T20401 C1V2RI 132353699 Ki = 35.8 nM T20401 C7Z4UB 132494202 Ki > 10000 nM T20401 CXN16P 132495328 Ki = 3.8 nM T20401 C20FGA 132495363 Ki > 500000 nM T20401 C4GR3Y 132498655 Ki = 0.48 nM T20401 CKLY32 132502995 Ki = 9533.7 nM T20401 CJQP17 132541861 Ki = 0.42 nM T20401 CVM1A9 132547283 Ki = 240 nM T20401 C3H1NS 132547284 Ki = 830 nM T20401 C1FWS2 132547285 Ki = 67.6 nM T20401 C7Z5LX 132547286 Ki = 368 nM T20401 CW97YT 132547287 Ki = 7.3 nM T20401 CW18RT 132547288 Ki = 18.1 nM T20401 COC54I 132547289 Ki = 22.3 nM T20401 CX4DM9 132547290 Ki = 19.5 nM T20401 C5JM7W 132547291 Ki = 15.1 nM T20401 C7V6XS 132547292 Ki = 13.2 nM T20401 C5O1JE 132547793 Ki > 100000 nM T20401 CKYC42 132547798 Ki = 59600 nM T20401 C7MZ8T 132569639 Ki = 590 nM T20401 CRL24F 132596304 Ki = 1480 nM T20401 C6OA8Z 132819872 Ki = 5.1 nM T20401 CJGH58 132819873 Ki = 9.3 nM T20401 COT92G 132819874 Ki = 3.7 nM T20401 COS36W 132819875 Ki = 2.9 nM T20401 CMAU69 132819876 Ki = 4.4 nM T20401 CY62CQ 132938107 Ki = 27.6 nM T20401 CB8T7K 132938108 Ki = 6.6 nM T20401 CY6L7Z 132941396 Ki = 22.4 nM T20401 C4K1YW 132961363 Ki = 2.4 nM T20401 CQ64ZM 132961364 Ki = 6 nM T20401 C5LGV6 132961365 Ki = 5.4 nM T20401 CD9ET2 132961426 Ki = 5 nM T20401 CR80OW 132961427 Ki = 85.4 nM T20401 C17QYW 132961557 Ki = 2.1 nM T20401 CGC58D 132961558 Ki = 9.1 nM T20401 CZDR23 132961559 Ki = 22.3 nM T20401 C4Y5SW 132961560 Ki = 3.2 nM T20401 CXF7N2 132961561 Ki = 2.5 nM T20401 CQAC41 132961562 Ki = 8.5 nM T20401 C57MKX 132961563 Ki = 8 nM T20401 C6N1PW 132961564 Ki = 17.4 nM T20401 CZ60IC 132961565 Ki = 8.4 nM T20401 CEP32W 132991412 Ki > 10000 nM T20401 C69NDK 133107891 Ki = 36.5 nM T20401 C2AIR8 134129901 Ki = 2.8 nM T20401 C1Y9AL 134130029 Ki = 0.97 nM T20401 CG0HL2 134130044 Ki = 56.2 nM T20401 C63CQL 134130121 Ki = 529 nM T20401 CU10DE 134130177 Ki = 20.1 nM T20401 C82HUT 134130285 Ki = 681 nM T20401 CMZ76O 134130322 Ki = 6350 nM T20401 CP8XK0 134130364 Ki = 3.4 nM T20401 C8AL2D 134130377 Ki = 244 nM T20401 C7N0JD 134130389 Ki = 301 nM T20401 C83LZE 134130471 Ki = 6.2 nM T20401 C5N8AO 134130483 Ki = 0.6 nM T20401 C9V3LX 134130512 Ki = 5.6 nM T20401 CO7G6J 134130566 Ki = 8.5 nM T20401 C69IZA 134130639 Ki > 10000 nM T20401 C8MGN3 134130817 Ki = 188.1 nM T20401 C52IRH 134131086 Ki = 2.1 nM T20401 CZ7CA3 134131127 Ki = 274 nM T20401 C9HVL2 134131189 Ki = 0.87 nM T20401 C5XU9Y 134131319 Ki = 3865 nM T20401 C7GBW5 134131361 Ki = 0.76 nM T20401 CZ2YK7 134131524 Ki = 2570 nM T20401 C3WJR8 134131535 Ki = 7.6 nM T20401 CQ0K5P 134131567 Ki = 1.6 nM T20401 C8Q5JZ 134131574 Ki = 163 nM T20401 CUVB06 134131580 Ki = 369 nM T20401 C94HZF 134131659 Ki = 0.83 nM T20401 CU5B8H 134131865 Ki = 1.5 nM T20401 CZQ3T2 134132041 Ki > 10000 nM T20401 C89TVU 134132755 Ki = 0.8 nM T20401 C2UIM6 134132835 Ki = 100.9 nM T20401 CECZ43 134133137 Ki > 500000 nM T20401 CFQG76 134133776 Ki = 49.3 nM T20401 CT8Z2Q 134133785 Ki = 8.6 nM T20401 C83QKJ 134133977 Ki = 1 nM T20401 CM3J9G 134134653 Ki = 24.3 nM T20401 CJ3EQ2 134136523 Ki = 2.6 nM T20401 CHR23F 134137004 Ki > 10000 nM T20401 C4IO1K 134137058 Ki = 20.1 nM T20401 C2X1UG 134137145 Ki = 8.2 nM T20401 CHM19B 134139215 Ki = 270.9 nM T20401 CWG0L5 134139228 Ki = 12.4 nM T20401 CRNF42 134140829 Ki = 58.3 nM T20401 C1T9JU 134140936 Ki = 883.4 nM T20401 CG4NU1 134141378 Ki = 5.4 nM T20401 CJ4R6E 134141819 Ki > 500000 nM T20401 CDUW03 134142004 Ki = 41.7 nM T20401 CC05JV 134142010 Ki = 13.2 nM T20401 CIK25S 134142323 Ki = 71.1 nM T20401 CIRG86 134142877 Ki = 4.4 nM T20401 CWT6O9 134142989 Ki = 6.3 nM T20401 C5BD1C 134143174 Ki > 10000 nM T20401 CWQ62J 134144541 Ki = 246.3 nM T20401 CG7X9K 134144756 Ki = 682.6 nM T20401 CJ5QD3 134144926 Ki = 1778.9 nM T20401 CR5F8T 134145685 Ki = 569 nM T20401 CBK73M 134146037 Ki = 4.3 nM T20401 C8FV5Y 134147016 Ki > 10000 nM T20401 C0TV9S 134147261 Ki = 9522 nM T20401 CDH38B 134147400 Ki = 15.7 nM T20401 CDSM29 134147656 Ki = 316 nM T20401 C85ABV 134147911 Ki = 350 nM T20401 CGBZ05 134148709 Ki = 61.5 nM T20401 CS7K8C 134149271 Ki = 150.7 nM T20401 C1Q8GK 134149666 Ki = 1.5 nM T20401 CF31OS 134149711 Ki = 31.6 nM T20401 CD5TI1 134149815 Ki = 297.3 nM T20401 CZ2C3J 134149835 Ki = 49 nM T20401 C2NXB7 134151324 Ki = 280 nM T20401 CIL4H9 134151823 Ki > 10000 nM T20401 C9GF7L 134152087 Ki = 4.6 nM T20401 CR4VE0 134152281 Ki > 500000 nM T20401 CU0T4X 134152542 Ki = 1.5 nM T20401 CZ9C1N 134152694 Ki = 24.1 nM T20401 CZ4WI8 134152920 Ki = 77.4 nM T20401 C4WBC6 134153047 Ki = 1.4 nM T20401 CD4EN0 134153199 Ki = 6809 nM T20401 CH6OT4 134153506 Ki = 6.6 nM T20401 CZ9T6I 134153525 Ki > 10000 nM T20401 CWSI54 134154346 Ki = 167.5 nM T20401 CSK6L9 134154625 Ki > 500000 nM T20401 CQZU97 134154945 Ki > 10000 nM T20401 CCU96S 134155195 Ki = 47.9 nM T20401 CG69UV 134155483 Ki > 500000 nM T20401 C52UTP 134156470 Ki = 0.5 nM T20401 C7OV6T 134156655 Ki = 426.1 nM T20401 CZ9L5F 134158397 Ki = 7.6 nM T20401 CR3Q5U 134159783 Ki = 7.6 nM T20401 CV9W6N 134159784 Ki = 6.3 nM T20401 C8C0TO 134812637 Ki = 8.2 nM T20401 CV9X5Y 134817795 Ki = 15.4 nM T20401 C19BHQ 134817796 Ki = 667.8 nM T20401 CY3E4D 134817797 Ki = 94.3 nM T20401 C8IF6V 134817798 Ki = 951.3 nM T20401 C0UL7A 134828600 Ki = 200 nM T20401 C4ZLP6 134828601 Ki = 270 nM T20401 C3OLP6 134828602 Ki = 210 nM T20401 CJT9W0 135393499 Ki = 0.5 nM T20401 CK8FP3 135393500 Ki = 0.6 nM T20401 CRL4V7 135393501 Ki = 0.5 nM T20401 C19SUQ 135405876 Ki > 10000 nM T20401 CTR37Z 135408753 Ki > 500000 nM T20401 C6QT0M 135411191 Ki = 120 nM T20401 C4TCL7 135411929 Ki = 523 nM T20401 C3YE2K 135412032 Ki > 10000 nM T20401 CW9B7C 135422576 Ki = 1.8 nM T20401 C4CXD1 135434964 Ki = 63.3 nM T20401 CFK9A4 135434965 Ki = 35.9 nM T20401 CY7RT4 135442220 Ki > 100000 nM T20401 CKAF26 135460193 Ki = 6.4 nM T20401 C1KUG5 135495066 Ki = 13100 nM T20401 C7E6AM 135496540 Ki = 250 nM T20401 C3MV2E 135519301 Ki = 9600 nM T20401 CPW4T3 135530880 Ki = 9.4 nM T20401 C0WEU9 135537166 Ki = 164 nM T20401 C7E8RX 135570228 IC50 = 9.33 nM T20401 C21GNK 135595335 Ki = 130.5 nM T20401 CC8IO3 135595465 Ki = 277 nM T20401 C74TBX 135595467 Ki = 365 nM T20401 C8D6XA 135595468 Ki = 12.6 nM T20401 CX1NF7 135595474 Ki = 413 nM T20401 CL71ND 135645043 Ki > 50000 nM T20401 CHM06N 135794287 Ki = 2150 nM T20401 C6J2RU 135878387 IC50 = 22 nM T20401 C1WH3Z 135891810 Ki = 7.6 nM T20401 CSH8M1 135995959 Ki = 5.5 nM T20401 CB90PQ 135995960 Ki = 8.3 nM T20401 C47ART 136002512 Ki = 170 nM T20401 C2J5FZ 136002546 IC50 = 450 nM T20401 CJ31YP 136002685 IC50 = 110 nM T20401 C0T8LG 136002686 Ki = 30 nM T20401 CXD6J2 136002687 IC50 = 80 nM T20401 CNG0L4 136044222 Ki = 707 nM T20401 CQ02AW 136044223 Ki > 10000 nM T20401 C47KQP 136053622 Ki = 264 nM T20401 C1M7DN 136053656 Ki = 690 nM T20401 C8CV0N 136056550 Ki = 43 nM T20401 CFT0H2 136059729 IC50 = 10 nM T20401 C31CEK 136094773 Ki = 0.53 nM T20401 C3VG8C 136094774 Ki = 4.4 nM T20401 C38LKD 136104491 Ki = 386000 nM T20401 C0PNH7 136104492 Ki = 7970 nM T20401 CNW21F 136104493 Ki = 3830 nM T20401 CST63W 136104494 Ki = 350000 nM T20401 C9GQS8 136104495 Ki = 8360 nM T20401 CHG82O 136118030 Ki = 12 nM T20401 C6RQS5 136123547 Ki = 51.5 nM T20401 C4O2IM 136123548 Ki = 79.7 nM T20401 C4KH2F 136138702 Ki = 31.1 nM T20401 C4A2XS 136198631 Ki = 12.95 nM T20401 C93PWB 136198632 Ki > 10000 nM T20401 CVME35 136198643 Ki = 619 nM T20401 CZ9M6L 136217534 Ki = 12.4 nM T20401 C8Q9ES 136217535 Ki = 259 nM T20401 CIX3N6 136217536 Ki = 349 nM T20401 CBO5I1 136242872 Ki = 5 nM T20401 CQDT25 136242873 Ki = 5.1 nM T20401 CK5AZ7 136242878 Ki = 6.1 nM T20401 C1NTA3 136418497 Ki = 167.7 nM T20401 CQUV48 136499038 Ki = 9.4 nM T20401 C6VS7N 136607460 Ki = 5.2 nM T20401 CAC75Q 136607461 Ki = 7.3 nM T20401 CYKW91 136728963 Ki = 41.4 nM T20401 CI28TM 136934908 Ki = 377 nM T20401 C9UKC8 136998786 Ki = 697 nM T20401 C3QFS1 136998787 Ki = 666 nM T20401 C1P9FJ 136998788 Ki = 596 nM T20401 CZ40LF 137028501 Ki = 11.8 nM T20401 C5Q8PD 137028502 Ki = 9.9 nM T20401 CSL47A 137028503 Ki = 6.4 nM T20401 C7T1HR 137028504 Ki = 5.9 nM T20401 C9WH2P 137028505 Ki = 4.3 nM T20401 CGBQ10 137028506 Ki = 4.6 nM T20401 C4DHG6 137028507 Ki = 5.5 nM T20401 CIP84X 137028508 Ki = 3.5 nM T20401 CF14KA 137028511 Ki = 31.3 nM T20401 CXHB30 137028512 Ki = 17.9 nM T20401 CRMC05 137028513 Ki = 2.9 nM T20401 CJH4E5 137028514 Ki = 3.8 nM T20401 CGAR93 137028515 Ki = 3.2 nM T20401 C4QG2K 137028516 Ki = 4.5 nM T20401 C2GMH5 137028517 Ki = 23.1 nM T20401 CBX6S7 137028518 Ki = 19.5 nM T20401 C52OFD 137028519 Ki = 565 nM T20401 CUW85H 137062187 Ki = 1645 nM T20401 C4XY9S 137091066 Ki = 157 nM T20401 C64ITR 137091070 Ki = 585 nM T20401 C0BEH8 137093138 Ki = 8.1 nM T20401 CD6C0A 137093141 Ki = 7.1 nM T20401 CJI35T 137124112 Ki = 428 nM T20401 CJI47D 137175023 Ki = 236 nM T20401 CM70RT 137175046 Ki = 618 nM T20401 CVZR36 137175050 Ki = 468 nM T20401 CCG5D7 137175057 Ki = 728 nM T20401 COFC53 137175058 Ki = 711 nM T20401 CV57WL 137175059 Ki = 652 nM T20401 CM1FL4 137175099 Ki = 309 nM T20401 CR6U9I 137175102 Ki = 547 nM T20401 CHK1L6 137175124 Ki = 683 nM T20401 CK2M1V 137175125 Ki = 264 nM T20401 CCP87O 137175126 Ki = 484 nM T20401 C4WZ5F 137175214 Ki = 454 nM T20401 CJ2DW1 137196867 Ki = 782.1 nM T20401 CUJ3N2 137196890 Ki = 425.6 nM T20401 CE9QV3 137226330 Ki = 7.1 nM T20401 C4SMA5 137226331 Ki = 7.6 nM T20401 C2H6VC 137226372 Ki > 10000 nM T20401 CZY9D7 137226374 Ki = 116 nM T20401 C6YBD3 137226375 Ki = 7.7 nM T20401 C7DMR8 137226384 Ki = 877 nM T20401 C2KG3D 137226385 Ki = 33 nM T20401 C0KMB4 137226399 Ki = 8.4 nM T20401 CD1VC9 137226400 Ki = 7.5 nM T20401 C4F8NU 137226401 Ki = 9.9 nM T20401 CW65FQ 137226402 Ki = 9.1 nM T20401 CY95JF 137226420 Ki = 14.5 nM T20401 CM58FB 137228156 Ki = 5.5 nM T20401 CK94PV 137228157 Ki = 7.1 nM T20401 CAY48F 137228158 Ki = 4.1 nM T20401 COW81G 137273278 Ki = 897 nM T20401 CY3P7J 137283379 Ki = 42.3 nM T20401 CPM09K 137287437 Ki = 55.43 nM T20401 CNS38T 137287438 Ki = 20.05 nM T20401 C1G8YE 137287439 Ki = 31.76 nM T20401 C1BOM7 137287440 Ki = 20.7 nM T20401 CY4K2R 137287441 Ki = 18.25 nM T20401 C39QNK 137287442 Ki = 52.17 nM T20401 CW52IQ 137631447 Ki = 4.44 nM T20401 CRK6Y9 137631731 Ki = 559.2 nM T20401 CZ5GQ4 137631746 Ki > 100 nM T20401 CFQ5W2 137631798 Ki = 26.3 nM T20401 CD47EX 137631815 IC50 = 198 nM T20401 CRHD41 137632004 IC50 = 0.855 nM T20401 C7O3CP 137632017 Ki = 12.14 nM T20401 C83VZC 137632115 Ki = 500 nM T20401 CBJ75C 137632178 Ki = 59.7 nM T20401 CN8UL1 137632214 Ki = 7.81 nM T20401 CYD0E3 137632442 Ki = 9.1 nM T20401 CWU67D 137632659 IC50 = 100 nM T20401 CL5K3D 137632743 Ki > 100 nM T20401 CE20FG 137632898 Ki = 24.23 nM T20401 CO25DP 137632949 Ki = 4 nM T20401 C9YKD5 137633039 Ki = 26.9 nM T20401 CFE79H 137633320 Ki > 10000 nM T20401 C5J3AX 137633409 Ki = 33.8 nM T20401 C9AD2H 137633797 Ki = 48.1 nM T20401 CVNO32 137633860 Ki = 28.1 nM T20401 C4CIT3 137634087 Ki = 1410 nM T20401 C5NLG4 137634142 Ki = 1750 nM T20401 CDF74L 137634370 IC50 = 10000 nM T20401 C7N0ER 137634525 Ki > 100000 nM T20401 C29PFJ 137634549 Ki = 1480 nM T20401 C0P6ZT 137634762 Ki = 68.6 nM T20401 CJT86I 137634882 IC50 = 65 nM T20401 CP0EC3 137635051 Ki = 272.4 nM T20401 C08ANJ 137635055 Ki = 860 nM T20401 CY1HI4 137635059 Ki = 77.2 nM T20401 C4YV1N 137635125 Ki = 687 nM T20401 C3NQ9Y 137635300 Ki = 89.9 nM T20401 C1ZKU2 137635320 Ki = 6.6 nM T20401 CZ1O5K 137635430 Ki = 3540 nM T20401 CS6M2N 137635469 Ki > 10000 nM T20401 CDB92Z 137635478 IC50 = 0.622 nM T20401 CNJV53 137635486 Ki = 1.21 nM T20401 CVNX12 137635652 Ki = 616 nM T20401 CZ4Q1T 137636083 Ki = 98.4 nM T20401 C9GIX7 137636130 Ki = 4.51 nM T20401 CV12YX 137636350 Ki > 100 nM T20401 CE46DY 137636432 Ki = 18.6 nM T20401 CK0N2Y 137636453 Ki = 79 nM T20401 C5R7LW 137636489 IC50 = 0.53 nM T20401 CM9YC2 137636494 Ki > 10000 nM T20401 CLR6U5 137636505 Ki = 79 nM T20401 C3PXL8 137636591 IC50 = 1.875 nM T20401 C5D3BS 137636775 Ki = 2030 nM T20401 CMX9T3 137636945 Ki = 7.62 nM T20401 CE9G5R 137636957 IC50 = 250 nM T20401 C7YKB0 137636981 Ki = 8.7 nM T20401 C2Z7GO 137637071 Ki = 16.9 nM T20401 C0H2CK 137637173 Ki = 24.6 nM T20401 CWI41E 137637209 IC50 = 500 nM T20401 CWO5Z6 137637365 Ki > 100 nM T20401 CGV9M8 137637508 Ki = 175.4 nM T20401 CG0N8K 137637564 Ki = 9.5 nM T20401 CDXW57 137637640 Ki = 340 nM T20401 CQ5K1H 137637688 Ki = 76.5 nM T20401 C80KCO 137637736 Ki = 157.4 nM T20401 C2HY8G 137637767 Ki = 16.9 nM T20401 CS3OY7 137638054 IC50 = 250 nM T20401 CPMN15 137638178 IC50 = 63 nM T20401 CB3KA0 137638304 Ki = 399.4 nM T20401 CHQ3P9 137638456 Ki = 6.8 nM T20401 CK6OW4 137638637 Ki = 4.8 nM T20401 C6V8ED 137638882 Ki = 4.9 nM T20401 C64JQN 137639095 Ki = 0.84 nM T20401 CVJ35I 137639180 Ki = 10.58 nM T20401 C12QYH 137639189 Ki = 1.14 nM T20401 C4LB2X 137639339 Ki = 66.9 nM T20401 CX7TE5 137639357 Ki = 735 nM T20401 C0IQ1U 137639377 Ki = 58.2 nM T20401 C29XAH 137639434 Ki = 9188.4 nM T20401 C8DW0G 137639460 IC50 = 0.802 nM T20401 CV4L6A 137639464 IC50 = 0.47 nM T20401 CH2C3F 137639611 Ki = 7.4 nM T20401 CPR04H 137639655 Ki = 126 nM T20401 C95ZIL 137639751 IC50 = 14000 nM T20401 C4SP7Q 137639785 Ki = 6.7 nM T20401 COE61G 137639833 Ki = 30900 nM T20401 C2OT9R 137640310 Ki = 0.69 nM T20401 C5OU2V 137640459 Ki = 177.3 nM T20401 CX3JI9 137640517 Ki = 8 nM T20401 CZGW35 137640627 Ki = 3650 nM T20401 CV1ZO5 137640742 IC50 = 290 nM T20401 CQN3L7 137640789 IC50 = 0.34 nM T20401 C8P3SC 137640892 Ki > 10000 nM T20401 CJ4M2A 137640917 Ki = 92.4 nM T20401 CR65OQ 137640944 Ki = 10 nM T20401 C75WMG 137641075 Ki = 265 nM T20401 C6B0CQ 137641198 Ki = 0.21 nM T20401 C0HER8 137641290 Ki = 8.8 nM T20401 CR2MU6 137641422 Ki = 16.31 nM T20401 CMOZ57 137641425 Ki = 9.1 nM T20401 C4FN0Q 137641666 Ki = 851 nM T20401 C53ZAF 137641717 Ki = 89.9 nM T20401 CR5JZ8 137642047 Ki > 10000 nM T20401 CCSN50 137642054 Ki > 100 nM T20401 CN6WS9 137642180 Ki = 43.2 nM T20401 C0Z9DH 137642233 Ki = 0.97 nM T20401 C6YV7B 137642310 Ki = 720 nM T20401 CEOC90 137642331 Ki = 861.1 nM T20401 CSY67B 137642513 Ki = 395.3 nM T20401 C51DEC 137642551 IC50 = 0.651 nM T20401 C8Z1YM 137642848 IC50 = 53 nM T20401 C61TSP 137642864 Ki > 100000 nM T20401 C7ZX8Q 137643203 Ki = 8.29 nM T20401 CKPG10 137643559 IC50 = 65 nM T20401 C3Y2GU 137643607 Ki = 28.9 nM T20401 C1BW5I 137643671 Ki = 5600 nM T20401 CN2M3C 137643724 Ki = 3430 nM T20401 CZ1W3N 137643790 IC50 = 0.799 nM T20401 C0B8QA 137643949 Ki > 100 nM T20401 CG13TO 137643998 Ki = 2.59 nM T20401 CF31BQ 137644307 Ki = 6.6 nM T20401 CI4A9L 137644641 Ki = 4660 nM T20401 CIK49D 137644678 Ki = 32.9 nM T20401 CV75NJ 137644865 Ki > 10000 nM T20401 CFA3R0 137644914 Ki = 302.1 nM T20401 CWQ91B 137644949 Ki = 19.8 nM T20401 CHG72J 137644957 Ki = 60.5 nM T20401 CM3DI7 137645052 IC50 = 202 nM T20401 CV0AH9 137645517 Ki = 203.1 nM T20401 C6UAB5 137645654 Ki = 17.8 nM T20401 CDZ6T8 137645734 Ki = 261.6 nM T20401 CFV6T3 137645790 Ki = 7.28 nM T20401 C3CI0M 137645793 Ki = 34.5 nM T20401 CBRK83 137645944 Ki = 9.5 nM T20401 C65SHT 137645986 IC50 = 250 nM T20401 C7E6NL 137646223 Ki = 4.3 nM T20401 C4WOE0 137646284 Ki = 426 nM T20401 C10YVU 137646329 Ki = 7.9 nM T20401 C5WG2P 137646543 Ki = 0.4 nM T20401 C0YFX2 137646956 Ki > 10000 nM T20401 C3AX0L 137647075 IC50 = 203 nM T20401 CVE3K2 137647149 IC50 = 0.287 nM T20401 CRP78K 137647221 Ki > 100 nM T20401 C5T2VN 137647270 Ki = 1580 nM T20401 CXD9A0 137647636 Ki = 0.29 nM T20401 CR2H7M 137647845 Ki = 5.2 nM T20401 CY15KD 137648125 Ki = 14 nM T20401 C5PEA6 137648128 Ki = 104 nM T20401 CCD71U 137648259 Ki = 6072.3 nM T20401 C49PLO 137648279 Ki = 761.9 nM T20401 CW8CL7 137648379 Ki = 3.9 nM T20401 CP2G0M 137648421 IC50 = 300 nM T20401 CU81DA 137648494 Ki = 65.4 nM T20401 CK14XO 137648525 Ki = 308.8 nM T20401 C21TVD 137648644 Ki = 197.1 nM T20401 C6RIM2 137648717 Ki = 63.9 nM T20401 C6IB1L 137648807 Ki = 551 nM T20401 C82NJP 137648964 Ki = 16.17 nM T20401 CEZT03 137649001 Ki = 20.3 nM T20401 CWP5O2 137649257 IC50 = 110 nM T20401 CI9LS2 137649321 Ki = 17.9 nM T20401 CY94BR 137649373 Ki = 2980 nM T20401 CSWR71 137649376 Ki = 48.3 nM T20401 C7PEQ0 137649468 IC50 = 0.41 nM T20401 CGLM50 137649870 Ki = 0.98 nM T20401 C2HA7Q 137649882 Ki > 10000 nM T20401 C4N1MP 137650156 Ki = 33.2 nM T20401 CCZ4N1 137650188 Ki = 9.2 nM T20401 C1FO3T 137650198 Ki = 1.1 nM T20401 C91KQA 137650256 Ki = 0.82 nM T20401 CD08YK 137650293 Ki = 21.8 nM T20401 CL9WK5 137650508 IC50 = 120 nM T20401 CKJ36G 137650647 Ki = 247.4 nM T20401 CD7S5L 137650698 Ki > 100000 nM T20401 CJV8Q6 137650823 Ki = 54.6 nM T20401 CBA5N4 137651134 IC50 = 45 nM T20401 CV89IF 137651491 Ki = 50.5 nM T20401 C5V6XP 137651635 Ki = 7 nM T20401 CSTP12 137651755 Ki = 3.2 nM T20401 C01BXO 137651769 Ki > 100 nM T20401 CRN60L 137651808 IC50 = 34 nM T20401 CBX26H 137652164 IC50 = 10000 nM T20401 CY0C6Z 137652226 Ki = 85.4 nM T20401 C6GWB1 137652305 Ki > 100 nM T20401 CN3RQ8 137652373 Ki > 10000 nM T20401 C5DG1K 137652445 Ki = 501 nM T20401 CP4GY0 137652940 Ki = 1710 nM T20401 C03TAW 137653117 Ki = 1190 nM T20401 CN0W6U 137653170 Ki > 50000 nM T20401 C9UGN4 137653309 Ki = 50.7 nM T20401 C45WNI 137653361 Ki = 3.24 nM T20401 C8Y7XR 137653485 Ki = 4.2 nM T20401 CIV3E9 137653528 Ki = 0.7 nM T20401 C4U9KA 137653686 Ki = 7.76 nM T20401 C0O3JI 137654169 Ki = 936 nM T20401 CKA95O 137654295 IC50 = 325 nM T20401 CTP0U2 137654343 Ki = 7.7 nM T20401 CNJ6P9 137654601 Ki > 10000 nM T20401 CS3LD8 137654917 Ki = 350 nM T20401 CRC23M 137655132 Ki = 122 nM T20401 CWT49Q 137655252 Ki = 504 nM T20401 CXC7I2 137655261 Ki = 34.4 nM T20401 C2P5FH 137655445 Ki = 27 nM T20401 C3DT7S 137655450 Ki > 100 nM T20401 CASB61 137655528 Ki > 100 nM T20401 C0XPN2 137655580 Ki = 295.6 nM T20401 CUO84H 137655694 Ki > 10000 nM T20401 CAZ27T 137655913 Ki = 7 nM T20401 C27ALW 137655946 Ki = 18.7 nM T20401 CC0OY9 137655984 Ki = 5.9 nM T20401 C8TJN9 137656061 Ki = 376.3 nM T20401 CJV27W 137656199 IC50 = 55 nM T20401 CHD58S 137656247 Ki > 10000 nM T20401 COEY05 137656447 Ki = 28.6 nM T20401 CRXD65 137656549 Ki = 7.22 nM T20401 C06ONV 137656670 Ki = 26.9 nM T20401 C0CK7G 137656796 Ki = 713.9 nM T20401 CG5EK0 137656938 Ki > 10000 nM T20401 CT7CW2 137657041 Ki = 1.42 nM T20401 C0ME2V 137657097 Ki = 4730 nM T20401 C3PAQ7 137657121 Ki > 10000 nM T20401 CM8UR7 137657283 IC50 = 210 nM T20401 C2SYC9 137657578 Ki = 82 nM T20401 C8RNZ6 137657759 Ki > 100 nM T20401 C0KI6G 137657917 Ki = 35.7 nM T20401 CTI2V7 137658103 Ki > 10000 nM T20401 CT5PO9 137658239 Ki = 3050 nM T20401 CH39CL 137658251 Ki = 10.7 nM T20401 C3W4BA 137658271 Ki = 23.2 nM T20401 C41MLN 137658275 Ki > 10000 nM T20401 CKX78V 137658314 Ki = 402.4 nM T20401 CL2H0T 137658375 Ki > 100 nM T20401 CTNZ72 137658510 IC50 = 25 nM T20401 CMR2L9 137658572 IC50 = 0.15 nM T20401 C7V6MY 137658589 Ki = 210 nM T20401 CT98MV 137658877 Ki > 100 nM T20401 C8YV5D 137659052 Ki = 0.28 nM T20401 CXO9Y7 137659205 Ki > 100 nM T20401 CE3VX9 137659225 IC50 = 0.39 nM T20401 CBS96V 137659241 IC50 = 7 nM T20401 CJ5O8M 137659269 Ki = 6.1 nM T20401 CO1RD4 137659342 Ki = 740 nM T20401 C5AM2K 137659383 Ki > 10000 nM T20401 C40MRZ 137659514 Ki = 4.85 nM T20401 CCX48V 137659570 Ki = 15.6 nM T20401 C9T2IO 137659737 IC50 = 5000 nM T20401 C4MB7C 137659778 Ki = 420 nM T20401 CXK83H 137659797 Ki = 6512.4 nM T20401 CHKB25 137659801 Ki > 10000 nM T20401 CSPB10 137659919 Ki = 32 nM T20401 C60DEN 137660288 Ki > 10000 nM T20401 CR45FV 137660495 IC50 = 232 nM T20401 CMS92X 137660799 Ki = 48.9 nM T20401 C0TZD5 137661006 Ki > 100000 nM T20401 C0PIE6 137661027 Ki = 67.6 nM T20401 CQ56MJ 137661167 Ki = 249.3 nM T20401 C62QWK 137661307 Ki = 94.2 nM T20401 CF6Z9A 137661353 Ki = 77.8 nM T20401 CRC92Y 137661359 Ki = 5.5 nM T20401 CN1JH4 137661469 Ki = 4.5 nM T20401 C1Z8KG 137661675 Ki = 3.5 nM T20401 C03HGD 137661687 IC50 = 0.19 nM T20401 C74YSR 137661914 Ki = 39.2 nM T20401 CEAR56 137662187 Ki = 7.9 nM T20401 CMP8S7 137662201 Ki = 14.9 nM T20401 CFR73V 137662256 Ki = 390.4 nM T20401 CO8UE3 137662293 Ki = 704.3 nM T20401 CTK0L9 137662315 IC50 = 0.338 nM T20401 C08ZTR 138393077 Ki = 1107.5 nM T20401 CIX41M 138393379 Ki = 0.7 nM T20401 C7V9ZF 138455154 Ki = 73.2 nM T20401 CBOM51 138753317 Ki = 1.2 nM T20401 CB83JY 139593608 Ki = 3.7 nM T20401 C8TWF0 139597735 Ki = 180 nM T20401 CR10ZH 139823666 Ki > 1000 nM T20401 C78UAW 142468585 Ki = 36.8 nM T20401 CZY8Q6 142468589 Ki = 1.1 nM T20401 C3HMI0 142468591 Ki = 151 nM T20401 CHA65U 142468595 Ki = 4050 nM T20401 C6KE9A 142468600 Ki = 3780 nM T20401 C65DHJ 142468602 Ki = 4.5 nM T20401 CI02LX 142468604 Ki = 242 nM T20401 C7LP3J 142468605 Ki > 50000 nM T20401 CA9O2I 142468608 Ki = 140 nM T20401 CUE58A 142547533 Ki > 10000 nM T20401 C6GB9T 143032987 Ki = 1566 nM T20401 CNW7H1 145948231 Ki = 3.9 nM T20401 C3PF4Q 145948234 Ki = 8.8 nM T20401 C7Y8GF 145949148 Ki = 276 nM T20401 CQC2D5 145949182 Ki = 83.4 nM T20401 C0Z2WP 145949184 Ki = 7 nM T20401 CI9H2E 145949226 Ki > 10000 nM T20401 CK65AC 145949290 Ki = 87 nM T20401 C8BZI0 145949366 Ki = 848.3 nM T20401 CP6AM5 145949377 Ki = 3 nM T20401 CHVR98 145949393 Ki = 920.8 nM T20401 CGLD54 145949403 Ki > 10000 nM T20401 C3LZH7 145949437 Ki = 17.7 nM T20401 CROP78 145949554 Ki = 16.1 nM T20401 C09ZGW 145949615 Ki = 889.2 nM T20401 CA01QK 145949650 Ki = 7.6 nM T20401 C7I3GC 145949670 Ki = 53.3 nM T20401 C7X0DZ 145949728 Ki = 364.6 nM T20401 CIU2Y1 145949743 Ki = 84.5 nM T20401 CA05JL 145949806 Ki = 48.9 nM T20401 CHI5L3 145949836 Ki = 6.8 nM T20401 C3U1AB 145949909 Ki = 67.3 nM T20401 C20RXT 145949974 Ki = 1.4 nM T20401 CJ8R3M 145950033 Ki = 176 nM T20401 CSW7B8 145950055 Ki > 10000 nM T20401 CISR74 145950124 Ki = 61.3 nM T20401 CRH3U4 145950259 Ki = 797 nM T20401 C7DBT4 145950298 Ki > 10000 nM T20401 CO9UN4 145950340 Ki = 35.8 nM T20401 CW56LV 145950373 Ki = 5.2 nM T20401 CJSK40 145950390 Ki > 10000 nM T20401 C2H9QY 145950512 Ki = 89.5 nM T20401 C7BK9O 145950527 Ki = 22 nM T20401 C63SMQ 145950568 Ki > 10000 nM T20401 CE58JF 145950709 Ki = 79.5 nM T20401 C0C9FT 145950755 Ki = 330.7 nM T20401 C0AC8O 145950774 IC50 = 27180 nM T20401 C8XAH1 145950880 Ki = 1.5 nM T20401 C53EGH 145950894 Ki = 1.2 nM T20401 CRD27H 145950965 Ki = 7.5 nM T20401 C8IGY9 145950981 Ki > 10000 nM T20401 C9QUL0 145951028 Ki = 0.51 nM T20401 C1X2FW 145951066 Ki = 1148 nM T20401 C7W5PI 145951214 Ki = 40.4 nM T20401 C87JIM 145951255 Ki = 155.5 nM T20401 CJ6LR3 145951259 Ki = 1253 nM T20401 CPD05I 145951366 Ki = 70.8 nM T20401 C7LMU1 145951380 Ki = 15 nM T20401 C86DBE 145951463 Ki = 376.5 nM T20401 CB8V7M 145951488 Ki = 55.4 nM T20401 CL25SI 145951508 Ki > 10000 nM T20401 CS8GO6 145951628 Ki = 1500 nM T20401 C38QHU 145951654 Ki = 61.7 nM T20401 CIM8X0 145951670 Ki = 4.9 nM T20401 CH9J8K 145951685 Ki = 8.3 nM T20401 C74RDJ 145951698 Ki = 59 nM T20401 CJ2W6V 145951720 Ki = 9.3 nM T20401 CZ23SB 145951758 Ki = 172 nM T20401 CC0P1U 145951787 Ki = 655.3 nM T20401 CN4MW7 145951794 Ki = 272 nM T20401 CF20QP 145951819 Ki = 6.2 nM T20401 C98SYV 145951855 Ki = 388.1 nM T20401 CQC79A 145951865 Ki = 48.9 nM T20401 C2OTU3 145951886 Ki = 0.94 nM T20401 CF7U3J 145951902 Ki = 91.6 nM T20401 CKZT53 145951931 Ki > 10000 nM T20401 C3R8NQ 145951979 Ki = 933.1 nM T20401 CGFU20 145952201 Ki > 10000 nM T20401 C4N3QL 145952239 Ki = 7.4 nM T20401 CUJ2G6 145952345 Ki = 14.1 nM T20401 CNDQ97 145952353 IC50 = 14100 nM T20401 CM30EN 145952365 Ki = 46.9 nM T20401 CU69PG 145952370 Ki = 94.7 nM T20401 C75RDX 145952490 Ki = 73.2 nM T20401 CP92AH 145952604 Ki = 59.7 nM T20401 C26OLK 145952634 Ki = 9.4 nM T20401 CW42HX 145952649 Ki = 14 nM T20401 C49OWE 145952696 Ki = 1547 nM T20401 C3ZR6A 145952729 IC50 = 36210 nM T20401 CWE6M8 145952775 Ki > 10000 nM T20401 C81UYG 145952794 Ki = 8.1 nM T20401 C6PZ3H 145952834 Ki = 67.1 nM T20401 CK4Q0X 145952846 Ki = 5.2 nM T20401 C56QVF 145952880 Ki = 8.8 nM T20401 CAS8M7 145952940 Ki = 703.2 nM T20401 CUB49H 145952983 Ki > 10000 nM T20401 CNZX07 145953044 Ki > 10000 nM T20401 C5M0RE 145953147 IC50 = 24320 nM T20401 C5C9RI 145953173 Ki = 431 nM T20401 C1KQ3D 145953178 Ki = 9.3 nM T20401 CZG27U 145953247 IC50 = 65220 nM T20401 CQM0J4 145953285 Ki = 7.9 nM T20401 C5DJY9 145953324 Ki = 15.9 nM T20401 CK5C4D 145953364 Ki = 841 nM T20401 CZO1Y8 145953466 Ki = 40.3 nM T20401 CFW94A 145953493 Ki = 6 nM T20401 CX37LN 145953547 Ki = 1838 nM T20401 C80OQZ 145953572 Ki = 31.1 nM T20401 C7Q4IN 145953662 Ki > 10000 nM T20401 C36ENH 145953837 Ki = 4.6 nM T20401 CH9N6D 145954010 Ki = 59.2 nM T20401 CVNE29 145954045 Ki = 6 nM T20401 C7GIQ5 145954093 Ki > 10000 nM T20401 CD52IH 145954185 Ki = 182.1 nM T20401 CM4U3B 145954289 Ki = 83.7 nM T20401 CZE24T 145954429 IC50 = 13500 nM T20401 C8R2HO 145954507 Ki = 2230 nM T20401 C7LZ1G 145954524 Ki = 65.7 nM T20401 C67HYG 145954632 Ki > 10000 nM T20401 CZG7I4 145954697 Ki = 6 nM T20401 CC08PM 145954740 Ki = 180.2 nM T20401 C0XO6A 145954770 Ki = 1.5 nM T20401 CTV8L5 145954775 Ki > 10000 nM T20401 CJ37XC 145954792 Ki = 1305 nM T20401 CNE86C 145954868 Ki = 7.7 nM T20401 C1LFA9 145954917 Ki = 90.2 nM T20401 CMZ2Y0 145954932 Ki = 0.85 nM T20401 C0UBV8 145955012 Ki = 16.6 nM T20401 C7QL4I 145955037 Ki = 38.8 nM T20401 C6UGK8 145955158 Ki = 30.7 nM T20401 CM9Y2S 145955268 Ki = 560 nM T20401 C0UG3K 145955383 Ki = 723.6 nM T20401 CHTR07 145955486 Ki = 32 nM T20401 CS6GA9 145955537 Ki = 8.6 nM T20401 C27JZH 145955576 Ki = 61.4 nM T20401 CW90OF 145955720 Ki = 59.3 nM T20401 CI64UX 145955888 Ki > 10000 nM T20401 CB86QZ 145955914 Ki = 199.6 nM T20401 CG7W8R 145955929 Ki = 38.9 nM T20401 CDWF95 145955978 Ki = 9.5 nM T20401 C9DLX6 145955997 Ki > 10000 nM T20401 CMGN62 145956070 Ki = 15.2 nM T20401 CS93JU 145956073 Ki = 44.1 nM T20401 CDJV68 145956076 Ki = 337.8 nM T20401 C5W1UM 145956081 Ki = 4209.2 nM T20401 CHXP91 145956144 Ki = 1.9 nM T20401 CZK0L8 145956164 Ki = 48.8 nM T20401 CY1AD2 145956169 Ki = 5.4 nM T20401 CD3LK5 145956229 Ki = 78 nM T20401 C89HDL 145956309 Ki = 4.9 nM T20401 CYJ3N0 145956346 Ki = 9.3 nM T20401 C2KV9S 145956347 Ki = 742.2 nM T20401 CQJO72 145956348 Ki > 10000 nM T20401 CGY39T 145956363 Ki = 80 nM T20401 CEL63H 145956491 Ki = 2 nM T20401 CAPD95 145956503 Ki > 10000 nM T20401 C4LH5W 145956563 Ki = 46 nM T20401 CRYP47 145956664 Ki > 10000 nM T20401 CE39IU 145956732 Ki > 10000 nM T20401 CYH7O8 145956770 Ki > 10000 nM T20401 CWPZ94 145956803 Ki = 0.54 nM T20401 CRUI17 145956819 Ki = 240.6 nM T20401 C6I1XE 145956976 Ki = 174.1 nM T20401 C7K2DA 145957040 Ki = 53.3 nM T20401 C7X6NA 145957099 Ki = 7.4 nM T20401 CEF41D 145957103 Ki = 234 nM T20401 CAMD59 145957136 Ki = 53.1 nM T20401 C94GRZ 145957236 Ki = 8.2 nM T20401 CED18K 145957307 Ki = 495.4 nM T20401 CC70NV 145957377 Ki > 10000 nM T20401 CKOX92 145957394 Ki = 326.2 nM T20401 C17FUI 145957430 Ki = 55.3 nM T20401 C6OR1Q 145957438 IC50 = 9100 nM T20401 CN5TM2 145957461 Ki = 358.6 nM T20401 C4S7BR 145957546 Ki = 74.2 nM T20401 C98PXC 145957555 Ki = 186.9 nM T20401 CL28OB 145957582 Ki = 756.2 nM T20401 CY37VB 145957610 IC50 = 38400 nM T20401 CP4TF7 145957664 Ki = 8.4 nM T20401 CI5B9M 145957665 Ki > 10000 nM T20401 C6HG7S 145957711 Ki = 48.6 nM T20401 CE4O0N 145957959 Ki = 38.9 nM T20401 CXFV43 145958041 Ki = 5.6 nM T20401 C3LZ9J 145958059 Ki = 1250 nM T20401 C6JL8X 145958066 Ki = 160.8 nM T20401 CM07ZF 145958200 Ki = 53 nM T20401 CQO8H5 145958250 Ki = 55.7 nM T20401 CJW72B 145958328 IC50 > 100000 nM T20401 CF07KV 145958447 Ki = 48.8 nM T20401 C5URQ2 145958565 Ki = 161 nM T20401 CC32ZJ 145958632 Ki = 1174.3 nM T20401 C0PRJ7 145958803 Ki = 52.5 nM T20401 C14UQR 145958824 Ki > 10000 nM T20401 C2MCO8 145958917 Ki > 10000 nM T20401 C0F9NS 145958940 Ki = 354.8 nM T20401 C52CMJ 145958993 Ki = 89 nM T20401 CUBA42 145958994 Ki = 94.8 nM T20401 CXVC18 145959110 Ki = 866.5 nM T20401 CNP7C0 145959116 Ki = 68.6 nM T20401 CU8J0M 145959118 Ki = 70.8 nM T20401 C1HML4 145959374 Ki = 327.8 nM T20401 C37CVT 145959395 Ki > 10000 nM T20401 C0LC9M 145959407 Ki = 4357.7 nM T20401 CGK4O1 145959409 Ki = 291.8 nM T20401 CM5OK6 145959413 Ki = 5.4 nM T20401 CWNS89 145959524 Ki = 41.2 nM T20401 C7J6MA 145959539 Ki > 10000 nM T20401 CJMU23 145959635 Ki = 61.9 nM T20401 CPL41Z 145959905 Ki = 4.4 nM T20401 CK8DX1 145959911 Ki > 10000 nM T20401 CGZ1K8 145959957 Ki = 14 nM T20401 C29YFS 145959974 Ki = 75 nM T20401 CL0NM5 145960039 Ki = 60.7 nM T20401 C9MSK2 145960116 Ki = 18.4 nM T20401 CH2K1A 145960207 Ki = 791.1 nM T20401 C2SI5J 145960220 Ki = 3.9 nM T20401 CB49ZJ 145960257 Ki > 10000 nM T20401 C6JND4 145960287 Ki = 0.18 nM T20401 C3JTG4 145960436 Ki = 450 nM T20401 C89GHI 145960779 Ki = 92.7 nM T20401 CVMF36 145960835 Ki = 327 nM T20401 CBGV25 145960853 Ki = 239 nM T20401 CT6U2G 145961010 Ki = 95.1 nM T20401 CD2X3F 145961133 Ki = 59 nM T20401 CBT85V 145961452 Ki = 277 nM T20401 C6JG2V 145961631 Ki = 69.9 nM T20401 CDA7G0 145962071 Ki = 33.4 nM T20401 CCYK28 145962259 Ki = 529 nM T20401 CQV18P 145962416 Ki = 485 nM T20401 C14OZY 145962693 Ki = 4.8 nM T20401 C34BRN 145962803 Ki = 571 nM T20401 C36LCF 145962935 Ki = 46.6 nM T20401 CZ9PL4 145963030 Ki = 158 nM T20401 CGY68S 145963294 Ki = 172 nM T20401 CJU15K 145963586 Ki = 120 nM T20401 CVL39I 145963679 Ki = 892 nM T20401 CUZ3A5 145963719 Ki = 293 nM T20401 C5VI0K 145964063 Ki = 7.9 nM T20401 CM71JT 145964104 Ki > 10000 nM T20401 CGTA80 145964130 Ki = 86.7 nM T20401 C9DE8Y 145964275 Ki = 6.1 nM T20401 C4C9IE 145964340 Ki = 7.4 nM T20401 CK21BE 145964400 Ki = 186.8 nM T20401 CAPU84 145964558 Ki = 6.1 nM T20401 C6FE1K 145964671 Ki = 57.6 nM T20401 CTC21S 145964779 Ki = 343.2 nM T20401 C3F4IS 145965133 Ki = 7.1 nM T20401 CGR16W 145965551 Ki = 760 nM T20401 C6RZT2 145965743 Ki = 38.4 nM T20401 CWHV36 145965762 Ki = 410 nM T20401 CINP09 145966173 Ki = 2.6 nM T20401 C2G8VU 145966250 Ki = 66.3 nM T20401 C5X7FM 145966343 Ki = 18.2 nM T20401 CCDI76 145966475 Ki = 25.2 nM T20401 CMF72D 145966553 Ki > 10000 nM T20401 CQ64RX 145966558 Ki = 5.4 nM T20401 CJ4D0R 145967030 Ki = 7 nM T20401 C7SUX3 145967040 Ki = 46.2 nM T20401 C7HZ6V 145967049 Ki = 69.6 nM T20401 CP8Q9U 145967308 Ki = 57.4 nM T20401 CFY3M6 145968026 Ki = 91.2 nM T20401 CDYR51 145968242 Ki = 78.8 nM T20401 C10PQH 145968245 Ki = 3.5 nM T20401 CKME70 145968701 Ki = 7.8 nM T20401 CX4D2R 145969379 Ki = 5 nM T20401 C9R4VB 145971458 Ki = 63.9 nM T20401 CD9I1U 145971467 Ki = 355.3 nM T20401 CZ71HS 145971486 Ki = 23 nM T20401 CC8D6E 145971537 IC50 = 29350 nM T20401 C73WMA 145971736 Ki = 51.3 nM T20401 C9P6UE 145971793 Ki = 416 nM T20401 C6DQK4 145972104 Ki = 47.1 nM T20401 CO4V1G 145972192 Ki = 32.3 nM T20401 CYMF38 145972316 Ki = 6.3 nM T20401 CP9H1U 145972366 Ki = 43.5 nM T20401 CD42QZ 145972397 Ki = 4.6 nM T20401 C93LTU 145972477 IC50 = 12100 nM T20401 CZ2LP7 145972551 Ki = 210.5 nM T20401 COJ6K4 145972603 Ki = 35.7 nM T20401 CS6D5R 145972711 IC50 = 14440 nM T20401 CGE23X 145972719 Ki = 220.5 nM T20401 CFXW14 145972912 Ki = 264.5 nM T20401 CF5KR4 145972986 Ki = 8.1 nM T20401 C65ZVF 145973004 Ki = 176.4 nM T20401 CN20BQ 145973308 Ki = 59.8 nM T20401 C1I8GK 145973355 Ki = 57.8 nM T20401 C9MZS1 145973465 Ki = 7.5 nM T20401 C8UAD6 145973595 Ki = 55.1 nM T20401 C7Y3WO 145973882 Ki = 4 nM T20401 C2C1KE 145973952 Ki = 8.3 nM T20401 CJ15WQ 145974101 Ki = 78.2 nM T20401 C7ZRI0 145974266 Ki = 23 nM T20401 CX5U8J 145974401 Ki = 5 nM T20401 CJD0I1 145974412 Ki = 4700 nM T20401 C2MF3Y 145974672 Ki = 4.4 nM T20401 C1QZ7F 145974710 Ki = 27.3 nM T20401 CG5SL1 145974949 Ki = 388.9 nM T20401 CVPA83 145974992 Ki = 6.3 nM T20401 CDU4M5 145975077 Ki = 6.7 nM T20401 C3I2WU 145975151 Ki = 43.7 nM T20401 C5U8RK 145975281 Ki = 598.2 nM T20401 C1VJD3 145975355 Ki = 466 nM T20401 CBL8Y4 145975424 Ki = 66.4 nM T20401 CT16KB 145975591 Ki = 1.8 nM T20401 CPK17Y 145975721 Ki = 530 nM T20401 CZVK21 145975933 Ki = 9.2 nM T20401 CQ08AT 145976207 Ki = 7.6 nM T20401 CO9M3B 145976300 Ki = 700 nM T20401 CI9C6U 145976539 Ki = 7.8 nM T20401 CZ7QU1 145976656 Ki = 4.5 nM T20401 C2BIZ4 145976658 Ki = 17.8 nM T20401 CHI26Q 145976735 Ki = 78.9 nM T20401 CZWC63 145977536 Ki = 4.2 nM T20401 CH3IC0 145977574 Ki = 24.3 nM T20401 CUEB47 145977814 Ki = 23.3 nM T20401 C81JIQ 145977869 Ki = 54.3 nM T20401 CL7GH8 145977904 Ki = 273.8 nM T20401 CK9L7E 145977947 Ki > 10000 nM T20401 C69UQY 145978025 Ki = 84.3 nM T20401 C5QSK0 145978140 Ki = 73.2 nM T20401 CO0J6L 145978583 Ki > 10000 nM T20401 CYG69V 145978605 Ki = 6.5 nM T20401 CYWK54 145978673 Ki = 284.7 nM T20401 C2D1TO 145978690 Ki = 506.6 nM T20401 CA32BT 145978780 Ki = 5.8 nM T20401 CXI41R 145978938 Ki = 860 nM T20401 CM8KP7 145979094 Ki = 530 nM T20401 C82LKO 145979169 Ki = 640 nM T20401 CI34JB 145979332 Ki = 94 nM T20401 CSPH69 145979414 Ki = 93.9 nM T20401 CQDB02 145979430 Ki = 559.1 nM T20401 CUDO01 145979473 Ki = 4590.8 nM T20401 COYX31 145979594 Ki = 373.2 nM T20401 CFUC92 145979600 Ki = 77 nM T20401 CXDE63 145979618 Ki = 260 nM T20401 C7ZOM8 145979619 Ki = 860 nM T20401 CIF72X 145979737 Ki = 4557.9 nM T20401 CMT6G7 145979772 Ki = 892.4 nM T20401 C8YA0B 145979831 Ki = 88.6 nM T20401 C5S9JX 145979949 Ki = 9.6 nM T20401 C9H6AW 145979979 Ki = 53 nM T20401 CLFJ74 145980146 Ki = 30.8 nM T20401 CD1IJ2 145980204 Ki = 9.8 nM T20401 CS85AP 145980216 Ki = 280 nM T20401 CWA24U 145980366 Ki = 488.1 nM T20401 CE3DP8 145980765 Ki = 80.4 nM T20401 C85TGI 145980938 Ki = 38.1 nM T20401 C97LPB 145981035 Ki = 465 nM T20401 C1RO4L 145981799 Ki = 460 nM T20401 C15PEL 145982039 Ki = 85.8 nM T20401 C4DNF7 145982126 Ki = 347.9 nM T20401 C7N6RT 145982437 Ki = 842.3 nM T20401 C2O8PK 145982576 Ki = 88.7 nM T20401 CK8MY4 145982622 Ki = 637.9 nM T20401 CX6Y5G 145982786 Ki = 27.2 nM T20401 C7M0HW 145982836 Ki = 91.5 nM T20401 C34LIQ 145982969 Ki = 707.8 nM T20401 CH3EF7 145983056 Ki = 406.3 nM T20401 CN7G5J 145983107 Ki = 807.5 nM T20401 C90VNX 145983131 Ki = 84.9 nM T20401 C9S0WG 145983404 Ki = 963.1 nM T20401 CWUJ59 145983568 Ki = 356.3 nM T20401 CB5G4W 145983664 Ki = 962.2 nM T20401 CF26VG 145983797 Ki = 92.6 nM T20401 C5SLN9 145983850 Ki = 48.9 nM T20401 CI52KO 145983856 Ki = 51.8 nM T20401 C3J5NQ 145983899 Ki = 95.1 nM T20401 C8PM9Y 145984067 Ki = 83.7 nM T20401 CA6I9T 145984095 Ki = 518.2 nM T20401 CEA52W 145984222 Ki = 66.2 nM T20401 CO9P3M 145984354 Ki = 53.3 nM T20401 C49ALP 145984517 Ki = 41 nM T20401 C8C0AB 145984626 Ki = 7524.5 nM T20401 CLDZ58 145984801 Ki = 459 nM T20401 C05FCU 145984802 Ki = 21.8 nM T20401 C7N6ZB 145984855 Ki = 730.7 nM T20401 C4FBS2 145985005 Ki = 553 nM T20401 CH8UK5 145985352 IC50 = 59 nM T20401 CZ8NA9 145985353 Ki = 29.6 nM T20401 C8Y1UT 145985534 Ki = 747.6 nM T20401 CF16KP 145985651 Ki = 245.1 nM T20401 CJEG52 145985679 Ki = 376.4 nM T20401 CN1WK4 145985761 Ki = 38.3 nM T20401 CIT98E 145985912 Ki = 666.3 nM T20401 C8VIF2 145985922 Ki = 51.6 nM T20401 CX0YW6 145985969 Ki = 71.3 nM T20401 C3E0RD 145986123 Ki = 57.1 nM T20401 CF7CH8 145986297 Ki = 559.5 nM T20401 CTZ71U 145986436 Ki = 1720 nM T20401 CIDO62 145986509 Ki = 450 nM T20401 CK05FT 145986641 Ki = 3080 nM T20401 CN56XE 145986933 Ki = 555.7 nM T20401 CG6CU5 145987209 Ki = 1647.7 nM T20401 CT01AM 145987366 Ki = 1810 nM T20401 C9UBE8 145987408 Ki = 7.7 nM T20401 CZPA17 145987454 Ki = 686.5 nM T20401 CI9F3V 145987533 Ki = 244.7 nM T20401 C65QOW 145987697 Ki = 29.6 nM T20401 CQF4O8 145987804 Ki = 784.1 nM T20401 CBF3V2 145987828 Ki = 771.7 nM T20401 C0LVN9 145987839 Ki = 598.6 nM T20401 C6RMF1 145987996 Ki = 9.5 nM T20401 C8XDH5 145988129 Ki = 2530 nM T20401 C89RFU 145988368 Ki = 79.7 nM T20401 CJ1P5W 145988462 Ki = 2792.7 nM T20401 CXA6F3 145988572 Ki = 84.8 nM T20401 CO3N6M 145988784 Ki = 3406.2 nM T20401 CPZN93 145988792 Ki = 565.1 nM T20401 CZW72V 145988876 Ki > 10000 nM T20401 C1LV0U 145988936 Ki = 8396.7 nM T20401 C39ZMI 145988963 Ki = 368.7 nM T20401 C7AUF1 145989028 Ki = 4416.5 nM T20401 C6BKP8 145989063 Ki = 840 nM T20401 C35VEG 145989087 Ki = 320 nM T20401 C6DN9E 145989219 Ki = 280 nM T20401 COZM89 145989422 Ki = 390 nM T20401 CJH51I 145989433 Ki = 3100 nM T20401 C9RVK0 145989853 Ki = 9385.9 nM T20401 CYJ79A 145989992 Ki = 186.7 nM T20401 CA8K2J 145990039 Ki = 160.9 nM T20401 C8XD2V 145990044 Ki = 2780 nM T20401 CLQ12A 145990129 Ki = 728.5 nM T20401 CHMR39 145990191 Ki = 413.6 nM T20401 CYOD69 145990290 Ki = 887.5 nM T20401 CZB2X3 145990392 Ki = 1447.5 nM T20401 CB63XC 145990519 Ki = 4131.1 nM T20401 CJQ73W 145990589 Ki = 530.3 nM T20401 C2WTN6 145990640 Ki = 595.9 nM T20401 CM6SA4 145990881 Ki = 1394.7 nM T20401 CIA37P 145991377 Ki = 1253.5 nM T20401 CWH89P 145991839 Ki = 2103.1 nM T20401 C3QXL4 145991981 Ki = 307.9 nM T20401 C9F8TL 145992666 Ki = 47.3 nM T20401 C58FGU 145992776 Ki = 4300 nM T20401 C7RYJ4 145992796 Ki = 822.3 nM T20401 CE34YK 145992956 Ki = 552.6 nM T20401 CH48GI 145992962 Ki = 997.6 nM T20401 CO42RK 145992983 Ki = 36.8 nM T20401 C8IE2X 145993014 Ki = 235.1 nM T20401 CDC84X 145993019 Ki = 7290.5 nM T20401 C7OZD6 145993265 Ki = 70.9 nM T20401 CE0HY6 145993300 Ki = 136.9 nM T20401 CS40WA 145993323 Ki = 67.9 nM T20401 CMS86X 145993352 Ki = 1900 nM T20401 CB12JK 145993432 Ki = 762.3 nM T20401 CZSC36 145993499 Ki = 76.2 nM T20401 CEC07M 145993642 Ki = 5150 nM T20401 CK3YT9 145993866 Ki = 74.6 nM T20401 CIDP76 145994238 Ki > 10000 nM T20401 C48CZD 146160385 Ki = 37.9 nM T20401 C2SG4L 146833326 Ki > 10000 nM T20401 C6FD2N 147348395 Ki = 3024 nM T20401 CGMX98 155510724 Ki = 0.08 nM T20401 C06MEW 155510831 Ki = 68.2 nM T20401 C3QJI5 155510851 Ki = 0.62 nM T20401 CY5T1K 155510897 Ki = 23.7 nM T20401 C1PG9M 155511036 Ki = 0.56 nM T20401 CN6DW9 155511075 Ki = 28.5 nM T20401 C2PXC3 155511133 Ki = 0.44 nM T20401 C1A5OB 155511232 Ki = 94.6 nM T20401 C30ADE 155511364 Ki = 651.4 nM T20401 C1D8JF 155511459 Ki > 10000 nM T20401 C6QNX5 155511723 Ki = 26.7 nM T20401 C03BJU 155511800 Ki = 60900 nM T20401 CJA94W 155512108 Ki = 0.64 nM T20401 CMCL94 155512138 Ki = 48.9 nM T20401 CE59ZG 155512211 Ki = 12.2 nM T20401 CI40CL 155512225 Ki = 4.3 nM T20401 C1ZPW3 155512418 Ki = 85.3 nM T20401 CQC04P 155512706 Ki = 525.2 nM T20401 C7J0HP 155512942 Ki = 67800 nM T20401 C51PHM 155512962 Ki > 10000 nM T20401 CN53ED 155512974 Ki = 77700 nM T20401 CLX19M 155512982 Ki = 0.48 nM T20401 CVSG61 155513076 Ki = 46.6 nM T20401 C21CAW 155513169 Ki = 40.6 nM T20401 CW1DP7 155513481 Ki = 6 nM T20401 C7QT4V 155513609 Ki > 10000 nM T20401 C5VT4X 155514082 Ki = 28.7 nM T20401 CX2UJ9 155514131 Ki = 64200 nM T20401 CZ5W1M 155514230 Ki = 273.1 nM T20401 CV7WR4 155514243 Ki = 8654 nM T20401 C67VGD 155514389 Ki = 0.38 nM T20401 CM5J3L 155514471 Ki = 19.8 nM T20401 CDM78Q 155514660 Ki = 4.6 nM T20401 C7W9NI 155514825 Ki = 647 nM T20401 CU9H2A 155514935 Ki = 9.7 nM T20401 CMQV46 155514970 Ki = 6.5 nM T20401 CCQB03 155515285 Ki = 3.9 nM T20401 CW08ZX 155515305 Ki = 44400 nM T20401 C5IPM8 155515308 Ki > 10000 nM T20401 C46UNX 155515514 Ki = 15.6 nM T20401 C6DG3E 155515525 Ki > 100000 nM T20401 C7MER6 155515557 Ki = 7100 nM T20401 C1C3SU 155515626 IC50 = 2600 nM T20401 C7UQ3J 155515746 Ki = 122 nM T20401 CT2ZB0 155515980 Ki = 0.6 nM T20401 C74SEH 155516204 Ki > 100000 nM T20401 CM9F7H 155516281 Ki = 295 nM T20401 CZN16J 155516304 Ki = 57.3 nM T20401 CLNT85 155516404 Ki = 46.8 nM T20401 COP4Q6 155516517 Ki = 20.7 nM T20401 C9LWV6 155516550 Ki = 0.35 nM T20401 C7IR3P 155516553 Ki = 18100 nM T20401 CBV6D3 155516701 Ki = 62.3 nM T20401 CP0NH3 155516885 Ki > 10000 nM T20401 C2E0ZF 155517026 Ki = 27.9 nM T20401 CAG9L4 155517430 Ki = 1.5 nM T20401 C3OW4N 155517544 Ki = 37.6 nM T20401 CW18JG 155517622 Ki = 56.7 nM T20401 C2H3JR 155517687 Ki > 100000 nM T20401 CQI20B 155517798 Ki > 100000 nM T20401 CRP2A6 155517861 Ki = 71.2 nM T20401 CWP3G6 155517862 Ki > 10000 nM T20401 CHA2R1 155517933 Ki = 84.3 nM T20401 CF07ZS 155517996 Ki = 0.68 nM T20401 C0O5CN 155518098 Ki > 10000 nM T20401 CUN49T 155518138 Ki = 70.5 nM T20401 C92QDE 155518180 Ki = 92.6 nM T20401 C1VNX3 155518220 Ki = 15.2 nM T20401 CP0U8D 155518225 Ki > 50000 nM T20401 CEH62Y 155518447 Ki = 5.9 nM T20401 CP7UI1 155518510 Ki = 12.8 nM T20401 CM7DQ6 155518807 Ki = 493.4 nM T20401 CHI59Y 155518875 Ki = 50400 nM T20401 CL92UI 155519026 Ki = 133.9 nM T20401 C5TO4Q 155519047 Ki > 100000 nM T20401 CRF95N 155519064 Ki = 86.3 nM T20401 CI84OL 155519083 IC50 = 140 nM T20401 CN8RC2 155519138 Ki = 592 nM T20401 CK21TJ 155519240 Ki = 22.9 nM T20401 C8MYG2 155519248 Ki = 3.6 nM T20401 CO6D1Y 155519288 Ki = 30.2 nM T20401 CC47MV 155519432 Ki = 94.4 nM T20401 CT56OD 155519473 Ki = 69.2 nM T20401 CI18TP 155519626 Ki = 230 nM T20401 CO4V0B 155519627 Ki = 4.4 nM T20401 CP4IL9 155519983 Ki = 24 nM T20401 CIV68R 155520019 Ki = 36.6 nM T20401 C5PN0D 155520029 Ki > 10000 nM T20401 C1AQP3 155520260 IC50 = 1620 nM T20401 CP49HE 155520274 Ki = 0.7 nM T20401 C4Z8MX 155520314 Ki = 86.9 nM T20401 C5JCL6 155520507 Ki > 10000 nM T20401 CG4VJ8 155520652 Ki = 0.05 nM T20401 C8E0SN 155520671 Ki = 61400 nM T20401 CE8QY5 155520792 Ki = 173.7 nM T20401 C4LPA1 155520806 Ki = 71.4 nM T20401 C80OQU 155520908 Ki = 340 nM T20401 CQ0OR1 155520930 Ki > 10000 nM T20401 CBM47H 155520952 Ki = 28.7 nM T20401 C9Z1FL 155521038 Ki > 10000 nM T20401 C2J1YG 155521041 Ki = 52.9 nM T20401 C2PR8W 155521294 Ki = 593.1 nM T20401 CN2X1Q 155521353 Ki = 25.7 nM T20401 CCGT71 155521462 Ki = 0.45 nM T20401 CB54YX 155521489 Ki = 9.3 nM T20401 CF7HE1 155521700 Ki = 1.6 nM T20401 CRQ4L3 155521766 Ki = 54.8 nM T20401 CZ7WI8 155521830 Ki = 5.6 nM T20401 CNP87G 155521876 Ki = 283.3 nM T20401 CR49AJ 155521885 Ki = 2.9 nM T20401 C4IYX7 155521930 Ki = 180.5 nM T20401 C2Q7BG 155522085 Ki = 223.4 nM T20401 C0A4EO 155522100 Ki = 11.1 nM T20401 CSN4C2 155522321 Ki = 215.7 nM T20401 C70NUX 155522372 Ki = 131.4 nM T20401 C8K9OI 155522618 Ki = 0.91 nM T20401 C6AWP0 155522679 Ki = 3.4 nM T20401 CDN9Z5 155522816 Ki = 1.4 nM T20401 C0Z3QT 155522883 Ki = 294 nM T20401 CJ49ZN 155522995 Ki = 5.3 nM T20401 CM3H1N 155523109 Ki = 3.3 nM T20401 CA9F2I 155523252 Ki = 5 nM T20401 C3HGK6 155523328 Ki = 2.4 nM T20401 C6YZM3 155523403 Ki = 77.3 nM T20401 C9Q2WR 155523406 Ki = 83.9 nM T20401 CWJ7R5 155523492 Ki = 2 nM T20401 CU2N9J 155523547 Ki = 1.5 nM T20401 CIF91M 155523572 Ki = 0.74 nM T20401 C8WP5K 155523621 Ki = 0.51 nM T20401 C9LF7B 155523634 Ki > 100000 nM T20401 C4U8XN 155523810 Ki = 194.7 nM T20401 CWD9Y1 155523853 Ki = 12.5 nM T20401 C3MX7F 155523857 Ki = 56.8 nM T20401 C0MZ5G 155524206 Ki = 0.44 nM T20401 C6KCG7 155524248 Ki = 139 nM T20401 CSC58M 155524279 Ki > 10000 nM T20401 CK86ZT 155524367 Ki = 9.5 nM T20401 CK80AQ 155524610 Ki = 90.1 nM T20401 C9PV5X 155524649 Ki = 94000 nM T20401 CS21YC 155524712 Ki = 2.6 nM T20401 CDO4X2 155524724 Ki = 86.4 nM T20401 C3DM5L 155524759 Ki = 503.4 nM T20401 C5J8AS 155524785 Ki = 52.7 nM T20401 CS0WP1 155524852 Ki = 265 nM T20401 C70ZPH 155524915 Ki = 2.9 nM T20401 C8M1KI 155525036 Ki = 71.6 nM T20401 CV6N0C 155525231 Ki = 9.6 nM T20401 CHT29F 155525313 Ki = 518.9 nM T20401 CPL80N 155525961 Ki = 28.7 nM T20401 CA02GS 155526086 Ki = 8.5 nM T20401 C4R1OT 155526288 Ki = 910 nM T20401 CGC8Y0 155526420 Ki > 10000 nM T20401 CKT14B 155526554 Ki > 10000 nM T20401 C0XZD3 155526695 Ki = 1460 nM T20401 C5JK0G 155526811 Ki = 0.75 nM T20401 CWGS97 155526825 Ki = 790 nM T20401 CGV91K 155527018 Ki = 9.5 nM T20401 CCL7V8 155527060 Ki = 92 nM T20401 CNVX86 155527078 Ki = 85.6 nM T20401 CAMY18 155527145 Ki = 0.61 nM T20401 CG8JZ9 155527153 Ki = 24.7 nM T20401 C8K3OI 155527167 Ki = 823.8 nM T20401 C1LDV0 155527209 Ki = 64.2 nM T20401 C1I5PO 155527240 Ki = 137 nM T20401 CK8XN6 155527284 Ki > 10000 nM T20401 C4N7OY 155527400 Ki = 92.1 nM T20401 CJ3K9W 155527428 Ki = 21.7 nM T20401 C4A5BC 155527483 Ki = 12.4 nM T20401 C7YW9E 155527622 Ki = 695 nM T20401 CDE96Y 155527673 Ki = 21.1 nM T20401 C65FOA 155527703 Ki = 611.5 nM T20401 C07LVI 155527781 Ki = 29.9 nM T20401 CPAH30 155527788 Ki = 57.9 nM T20401 C5XC7V 155527967 Ki = 7608 nM T20401 CDN05K 155527975 Ki = 0.91 nM T20401 C0RJ2M 155528294 Ki = 95.4 nM T20401 CN9G0E 155528332 Ki = 184 nM T20401 C4IML7 155528345 Ki = 75.1 nM T20401 CLF2V0 155528496 Ki = 153.8 nM T20401 C38SKR 155528605 Ki = 40.6 nM T20401 CB08MU 155528753 Ki = 75700 nM T20401 C2LF1H 155528761 Ki = 34.9 nM T20401 C5X0CS 155528825 Ki > 100000 nM T20401 CN27OU 155528858 Ki = 2660.2 nM T20401 C7DCG0 155529026 Ki = 73.1 nM T20401 CECZ45 155529036 Ki = 932.9 nM T20401 C1T2EA 155529101 Ki = 74.2 nM T20401 CWEQ38 155529122 Ki = 20.5 nM T20401 C52QUD 155529352 Ki = 29.5 nM T20401 C8DN2F 155529373 Ki = 32.6 nM T20401 CG94RZ 155529376 Ki = 605.8 nM T20401 C2HUS1 155529422 IC50 = 15.97 nM T20401 C6TQ7W 155529566 IC50 = 5820 nM T20401 C2NY1E 155529877 Ki > 2000 nM T20401 C2JV7R 155529885 Ki = 342 nM T20401 CG3J0Q 155529984 Ki = 9103.9 nM T20401 CJ21OD 155530289 Ki > 50000 nM T20401 CW07EO 155530326 Ki = 47 nM T20401 CKO2V5 155530358 Ki = 56.4 nM T20401 C7TV5H 155530408 Ki = 7.4 nM T20401 CIGQ50 155530440 Ki = 8.7 nM T20401 C9Y4VC 155530502 Ki = 1.3 nM T20401 CTJ3I7 155530506 Ki = 22.8 nM T20401 C0HQ8E 155530537 Ki = 22.2 nM T20401 CP3UJ0 155530687 Ki = 0.93 nM T20401 C2T0LQ 155530848 Ki = 44.5 nM T20401 C3GK9H 155530900 Ki = 12 nM T20401 C2MT3K 155530925 Ki = 27.5 nM T20401 C2X1JQ 155530996 Ki = 5.5 nM T20401 COY7L3 155531072 Ki = 92.1 nM T20401 C8C4BT 155531090 Ki = 142 nM T20401 CICU68 155531183 Ki = 2106 nM T20401 CGN43T 155531186 Ki > 2000 nM T20401 CO7P5W 155531268 Ki = 0.6 nM T20401 CLMZ93 155531382 Ki = 1.7 nM T20401 CYBD02 155531537 Ki = 3930 nM T20401 C43LZI 155531630 Ki = 8.9 nM T20401 CC5L6V 155531813 Ki = 35 nM T20401 CFV23M 155531820 Ki > 100000 nM T20401 CW6TC5 155531936 Ki = 48400 nM T20401 CUM2B8 155532026 Ki = 9300 nM T20401 C83DJY 155532441 Ki > 100000 nM T20401 CASV53 155532466 Ki = 75 nM T20401 CFK8R5 155532512 Ki > 100000 nM T20401 CH6QB8 155532578 IC50 = 3300 nM T20401 CQ0XM6 155532587 Ki = 597.7 nM T20401 C5H8QF 155532861 Ki = 744.5 nM T20401 CG7Y5M 155532951 Ki = 69640 nM T20401 CKY1I8 155533416 Ki = 60.5 nM T20401 CDM2Y1 155533454 Ki = 0.59 nM T20401 C64XYO 155533459 Ki = 0.72 nM T20401 C0BNY7 155533528 Ki = 37.3 nM T20401 CPX2T1 155533590 Ki = 81.8 nM T20401 COK37H 155533887 Ki = 360 nM T20401 CTKI39 155533898 Ki = 903.6 nM T20401 C3FAC0 155533901 IC50 = 310 nM T20401 C0I5XS 155534055 Ki = 2.1 nM T20401 C78ZFI 155534074 Ki = 4.4 nM T20401 CT5NG1 155534179 Ki = 19.6 nM T20401 CPG13Y 155534247 Ki = 65.5 nM T20401 C6UF3R 155534332 Ki > 10000 nM T20401 CR2A6J 155534340 Ki = 6945 nM T20401 C14TGQ 155534675 Ki = 14.7 nM T20401 CS0FK9 155534753 Ki = 3.8 nM T20401 CK4TR2 155534861 Ki > 10000 nM T20401 CS5OI9 155534862 Ki = 8.9 nM T20401 CHG10E 155534912 Ki = 0.67 nM T20401 C67ROE 155534951 Ki = 28.7 nM T20401 C0QW8K 155535058 Ki = 13.2 nM T20401 CE1I8S 155535343 Ki = 3925 nM T20401 CC7M4N 155535347 Ki = 307.7 nM T20401 CVU5P6 155535355 Ki = 0.8 nM T20401 CV0N9I 155535382 Ki > 10000 nM T20401 CKR07J 155535598 Ki = 370.5 nM T20401 CNFR72 155535756 Ki = 56300 nM T20401 CFYA23 155535780 Ki = 7.8 nM T20401 CD2O3A 155535852 Ki = 908 nM T20401 CLJ64Q 155535889 Ki = 38 nM T20401 CZPY79 155536184 Ki = 90 nM T20401 CF0PC4 155536422 Ki > 10000 nM T20401 CW92OP 155536652 Ki = 9.9 nM T20401 CB47KF 155536691 Ki = 440.1 nM T20401 C0EDQ2 155536876 Ki = 65 nM T20401 CZ0T6A 155537018 Ki = 483.6 nM T20401 COP2R4 155537042 Ki = 44.8 nM T20401 C6T7BQ 155537167 Ki = 2275 nM T20401 C1K9AC 155537404 Ki > 10000 nM T20401 CXQ23T 155537493 Ki > 100000 nM T20401 C4K0MB 155537772 Ki = 3300 nM T20401 C0CG6Q 155537790 Ki = 42.2 nM T20401 C47OHJ 155537809 Ki = 15.6 nM T20401 C67ZET 155537843 Ki = 9.6 nM T20401 CYM0A3 155538069 Ki = 6.7 nM T20401 C5RV9W 155538073 Ki = 4.9 nM T20401 COX74J 155538083 Ki = 4.8 nM T20401 C60IZQ 155538189 Ki = 82.9 nM T20401 CB2EI4 155538212 Ki = 57.7 nM T20401 C9AP8F 155538224 Ki = 26.2 nM T20401 CB8C4X 155538289 Ki = 7700 nM T20401 C13GKU 155538478 IC50 = 1320 nM T20401 C3XSM6 155538611 Ki = 267.8 nM T20401 CM6D1H 155538676 Ki = 35.4 nM T20401 CHQP36 155539441 Ki = 44.3 nM T20401 CKE72Y 155539552 Ki = 0.82 nM T20401 C94OZU 155539579 Ki = 438.7 nM T20401 C9K2TL 155539730 Ki = 5.2 nM T20401 CS1G5V 155539783 Ki = 64.8 nM T20401 CS1UR7 155539868 Ki = 61.7 nM T20401 C85YWZ 155539989 Ki = 182.3 nM T20401 C53TKA 155540088 Ki = 43.6 nM T20401 CSAD81 155540401 Ki = 17.5 nM T20401 CZ8FJ3 155540422 Ki = 4.5 nM T20401 CW9B0X 155540441 Ki > 10000 nM T20401 C2VAD8 155540596 Ki = 0.69 nM T20401 C95TBC 155540629 Ki = 2.2 nM T20401 CCO34J 155540665 Ki > 10000 nM T20401 CGNS87 155540756 Ki = 0.88 nM T20401 CFN03K 155540920 Ki = 41.5 nM T20401 CGVJ81 155540983 IC50 = 500 nM T20401 C4H1ZC 155541040 Ki = 28.3 nM T20401 C3CLU2 155541078 Ki > 2000 nM T20401 C7Z6FC 155541724 Ki > 10000 nM T20401 C8RV6T 155541805 Ki = 47.1 nM T20401 CW96ES 155541807 Ki = 0.78 nM T20401 C4MW9Q 155541811 Ki = 56.4 nM T20401 C5F3SJ 155541888 Ki = 27.6 nM T20401 CX20DK 155541945 Ki = 1714 nM T20401 CZ2CT0 155542259 Ki = 6020 nM T20401 CW61DF 155542555 Ki = 34.8 nM T20401 CA75HO 155542580 Ki = 8.9 nM T20401 CTL8O3 155542606 Ki = 45.9 nM T20401 C3RC8T 155542635 Ki = 34.5 nM T20401 CT9GZ2 155542660 Ki = 262.1 nM T20401 CDK2W5 155542691 Ki = 9.5 nM T20401 CA76LB 155542698 Ki = 7500 nM T20401 CY3BO6 155542934 Ki = 53.5 nM T20401 C75TVG 155542954 Ki = 8.5 nM T20401 C2AEH6 155543096 Ki = 411 nM T20401 CN2SJ7 155543228 Ki = 38.2 nM T20401 C19DJA 155543271 Ki = 4.3 nM T20401 CHKV89 155543295 Ki = 4.3 nM T20401 CRF64E 155543422 Ki = 89.5 nM T20401 CLF3N5 155543891 Ki = 0.29 nM T20401 CPV20B 155543950 Ki = 9.3 nM T20401 C08DHT 155544006 Ki > 10000 nM T20401 C30HST 155544165 Ki = 44.8 nM T20401 CN0E1V 155544321 Ki = 43 nM T20401 CS9WR6 155544336 Ki > 2000 nM T20401 C7PC5J 155544382 Ki = 0.03 nM T20401 CSX2H7 155544608 Ki = 536.9 nM T20401 CGP7Z0 155544629 IC50 = 2100 nM T20401 CI2T8N 155544664 Ki = 4.8 nM T20401 CRM69J 155544710 Ki = 5.3 nM T20401 CP27AW 155544846 Ki > 10000 nM T20401 CDXL09 155544901 Ki = 7.2 nM T20401 C0BV1J 155545536 Ki = 56.9 nM T20401 CQV78W 155545657 Ki = 126.6 nM T20401 CB6J9G 155545674 Ki > 10000 nM T20401 CY6SX5 155545800 Ki = 44200 nM T20401 CP2SZ7 155545812 Ki = 4350 nM T20401 C95IJM 155545916 Ki = 541 nM T20401 C3Y8LT 155546146 Ki = 28.7 nM T20401 C9M2FW 155546556 IC50 = 1210 nM T20401 CG0E1W 155546684 IC50 = 1230 nM T20401 CSW62L 155546892 Ki = 39300 nM T20401 CC4IG8 155547081 Ki = 28.7 nM T20401 CF3UL5 155547275 Ki = 0.42 nM T20401 CV7OB5 155547342 Ki > 100000 nM T20401 C9E2KH 155547486 Ki = 81.4 nM T20401 C59MDT 155547507 Ki = 19.9 nM T20401 C83ZIS 155547526 Ki = 11.4 nM T20401 CW19PC 155547551 Ki = 589 nM T20401 C73YLV 155547628 Ki = 0.62 nM T20401 C9FVY6 155547723 Ki = 19.5 nM T20401 C61MSB 155547730 Ki = 0.42 nM T20401 CK5UD3 155547819 Ki = 13.2 nM T20401 CP4N3X 155547901 Ki = 4.4 nM T20401 CU94YA 155548070 Ki = 43.7 nM T20401 CCUN29 155548118 Ki > 10000 nM T20401 C3IO2B 155548134 Ki > 10000 nM T20401 C3JYG2 155548272 Ki = 870.9 nM T20401 CQG5F9 155548326 Ki = 34.9 nM T20401 C6XBZ3 155548352 Ki = 0.78 nM T20401 CUTY40 155548640 Ki = 262.3 nM T20401 CH2KB7 155548697 Ki = 20.8 nM T20401 CN7S5W 155548866 Ki = 10.9 nM T20401 CDC0F4 155548911 Ki = 27.3 nM T20401 CU1NE7 155549031 Ki = 0.7 nM T20401 C9JOV3 155549090 Ki = 0.72 nM T20401 CA25QH 155549266 Ki = 18.4 nM T20401 CR79SY 155549354 Ki = 6880 nM T20401 CL2B4T 155549378 Ki = 3.5 nM T20401 C6PY2G 155549478 Ki = 0.45 nM T20401 C2CLU0 155549558 Ki = 65.2 nM T20401 CIG6A7 155549616 Ki = 6.9 nM T20401 C1JR2F 155549662 Ki = 6493 nM T20401 CF6CW3 155549677 Ki = 83.3 nM T20401 C8NS5F 155549723 Ki = 908 nM T20401 CEZX49 155549753 Ki = 8.9 nM T20401 C8GZK4 155549788 Ki > 100000 nM T20401 CAYO49 155550021 Ki = 32.7 nM T20401 C3YN0W 155550099 Ki = 65.7 nM T20401 C1ZMC2 155550117 IC50 = 1490 nM T20401 CZB57Y 155550558 Ki = 0.06 nM T20401 CHO96B 155550610 Ki = 24300 nM T20401 C4O6TN 155550616 Ki = 9.1 nM T20401 CMWQ79 155550618 Ki = 71.5 nM T20401 C6XPV0 155550626 Ki = 5.2 nM T20401 CB2Q4M 155550927 Ki = 77.3 nM T20401 CG0MQ3 155551020 Ki = 0.07 nM T20401 CTE04H 155551088 Ki = 2344 nM T20401 CPRC19 155551316 Ki = 0.54 nM T20401 C4S0JZ 155551334 Ki = 234.1 nM T20401 CL2H8V 155551536 Ki = 39200 nM T20401 CSY39H 155551651 Ki = 160 nM T20401 C69AYQ 155551705 Ki > 100000 nM T20401 COC4Z9 155551784 Ki = 17.9 nM T20401 CZ0T3C 155551786 Ki = 4 nM T20401 C3AN2K 155551935 Ki = 2581 nM T20401 CG9PN8 155552113 Ki = 5.8 nM T20401 C7E3UF 155552316 Ki = 6200 nM T20401 C3DHB7 155552411 Ki = 6470 nM T20401 CW8S7L 155552594 Ki = 30 nM T20401 CZ6VL4 155552603 Ki = 28.7 nM T20401 CN25FV 155552708 Ki = 13.1 nM T20401 CBQ42J 155552773 Ki = 45000 nM T20401 CFT82G 155552780 Ki = 107.5 nM T20401 C0OG8P 155553361 Ki = 0.24 nM T20401 CP15VC 155553400 Ki = 593 nM T20401 CYS29E 155553445 Ki = 4440 nM T20401 C1QJ3H 155553542 Ki = 51.5 nM T20401 C82WXR 155553544 Ki = 869.6 nM T20401 CQM27S 155553591 Ki = 66.6 nM T20401 CQ1PE4 155553611 Ki > 100000 nM T20401 C1R7CJ 155553759 Ki = 3.7 nM T20401 C02LSY 155553787 Ki > 10000 nM T20401 C2J3ZT 155553989 IC50 = 1300 nM T20401 C8SO9P 155554095 Ki = 44.3 nM T20401 C6IMR3 155554140 Ki = 0.87 nM T20401 CMEP40 155554179 Ki = 7.9 nM T20401 CE57CO 155554263 Ki = 254 nM T20401 C0U8CG 155554286 Ki = 212.9 nM T20401 C6D9BJ 155554303 Ki > 10000 nM T20401 C3W6RT 155554309 Ki = 1680 nM T20401 C7VMB9 155554430 IC50 = 1040 nM T20401 CNX5L2 155554533 Ki = 77.8 nM T20401 C5VLU4 155554670 Ki = 439.8 nM T20401 CM4I0O 155554763 Ki = 55800 nM T20401 CZU9Y7 155554800 Ki = 6.9 nM T20401 CW5F4A 155554840 Ki = 97.8 nM T20401 CA78FQ 155555070 Ki = 5310 nM T20401 C5YA7C 155555084 Ki = 13.3 nM T20401 C9W1ET 155555489 Ki > 10000 nM T20401 CJ06PN 155555584 Ki = 1950 nM T20401 CV2NZ0 155555718 Ki = 138.6 nM T20401 CUY2C6 155555751 Ki = 0.39 nM T20401 CA7UK2 155555803 Ki = 31.5 nM T20401 CXNZ49 155555817 Ki = 1.7 nM T20401 CX4P1W 155555874 Ki = 456.2 nM T20401 CWB82E 155555878 Ki = 0.71 nM T20401 CKIR52 155556062 Ki = 20.1 nM T20401 C9I0QN 155556147 Ki = 28.7 nM T20401 CN9IJ3 155556148 IC50 = 410 nM T20401 C84MNE 155556163 Ki = 42.8 nM T20401 C5PZF2 155556257 Ki = 94.2 nM T20401 CM60WT 155556386 Ki = 74.7 nM T20401 CD4K6H 155556521 Ki = 0.7 nM T20401 CVR2X5 155556659 Ki > 100000 nM T20401 CGZ58Y 155556761 Ki = 16.9 nM T20401 C2Q3UO 155556889 Ki = 858.3 nM T20401 CYZ3K0 155556908 Ki = 6.9 nM T20401 CG8L0O 155557058 Ki = 15.9 nM T20401 CHKA19 155557282 Ki = 4.8 nM T20401 CJF9O7 155557300 Ki = 92000 nM T20401 C87GRH 155557329 Ki = 526.1 nM T20401 CRK5I0 155557428 Ki = 289 nM T20401 C40MOH 155557452 Ki = 0.36 nM T20401 C1RMC6 155557757 Ki = 5034 nM T20401 CNX9J2 155557875 Ki = 9 nM T20401 CM6NU0 155557925 Ki = 9.8 nM T20401 CWK35T 155557969 Ki = 8.8 nM T20401 CQI5Z4 155558076 Ki = 629.6 nM T20401 CK8GH2 155558119 Ki = 0.3 nM T20401 CME2Z4 155558216 Ki = 3.2 nM T20401 C70WSB 155558230 Ki > 10000 nM T20401 C52RLU 155558376 IC50 = 1600 nM T20401 CQ2ML6 155558561 Ki = 479 nM T20401 CK1RO0 155558641 Ki = 0.64 nM T20401 CH1Z2S 155558695 Ki = 7600 nM T20401 C4V2PS 155558747 Ki = 6.5 nM T20401 C6QXP8 155558748 Ki = 7270 nM T20401 CZ7C0S 155558990 Ki = 8 nM T20401 CI2XS3 155559081 Ki = 8.5 nM T20401 CGQ7S0 155559325 Ki = 3.6 nM T20401 C6CY3G 155559512 Ki = 0.09 nM T20401 CNT0F5 155559682 Ki > 10000 nM T20401 CK7H8I 155559761 Ki = 16.5 nM T20401 C3Y7WJ 155560101 Ki = 53400 nM T20401 CZ2A7O 155560148 Ki = 270.5 nM T20401 CB2X0V 155560428 Ki = 2580 nM T20401 CB5S8V 155560635 Ki = 78.6 nM T20401 COC45S 155560702 Ki = 221.5 nM T20401 CY1TF7 155560798 Ki = 0.08 nM T20401 C0U1NP 155560951 Ki = 3.5 nM T20401 CFY9A2 155561027 Ki = 207 nM T20401 CP3H0R 155561119 Ki = 78200 nM T20401 C3FG8W 155561198 Ki = 2900 nM T20401 CSK5X2 155561354 Ki > 10000 nM T20401 C2SZM0 155561361 Ki = 39.4 nM T20401 CHA8R0 155561556 Ki = 28.7 nM T20401 CAP5I4 155561568 Ki = 0.83 nM T20401 CU03LF 155561751 Ki = 134.6 nM T20401 CY9N4P 155561775 Ki = 2300 nM T20401 CU1JV7 155561839 Ki = 540.9 nM T20401 CJ5Y6X 155561851 Ki = 2154 nM T20401 CXE2R9 155561928 Ki = 36.2 nM T20401 C5W7MQ 155562360 Ki = 62.3 nM T20401 CG43PS 155562766 Ki = 25 nM T20401 C2FW8S 155562815 Ki = 8.2 nM T20401 CJ74ND 155563017 Ki = 12.6 nM T20401 C1J3UH 155563153 Ki = 97400 nM T20401 C7A8EX 155563186 Ki = 246.4 nM T20401 C9SH6R 155563203 Ki = 63300 nM T20401 C6KD7C 155563215 Ki = 52.2 nM T20401 CP85AZ 155563623 Ki = 26.3 nM T20401 C89MTB 155563810 Ki = 2084 nM T20401 C0GU6P 155563888 Ki = 692.2 nM T20401 CQ40DU 155563908 Ki = 339 nM T20401 C2XB6V 155564028 Ki = 826.3 nM T20401 CF7XH2 155564101 Ki = 94.2 nM T20401 CGY32K 155564210 Ki = 460.4 nM T20401 CY9M4F 155564463 Ki = 4670 nM T20401 C97TMY 155564559 Ki = 339 nM T20401 C1K0LR 155564617 Ki = 53.9 nM T20401 C07GFY 155564664 Ki = 7.9 nM T20401 CY9IW2 155564942 Ki = 0.55 nM T20401 CNV35X 155565135 Ki = 25.4 nM T20401 C0XO6Z 155565139 Ki > 10000 nM T20401 C0E4QV 155565149 Ki = 3 nM T20401 C5XV7O 155565283 Ki = 0.04 nM T20401 CNL8B7 155565372 Ki = 5761.4 nM T20401 CI5MV1 155565395 Ki = 114.9 nM T20401 CJ7I6Z 155565419 Ki = 3.2 nM T20401 CDF5E6 155565628 Ki = 9443 nM T20401 C0COK6 155565635 Ki = 837.6 nM T20401 CT9Z5H 155565773 Ki = 1750 nM T20401 CW3N9Z 155566095 Ki = 383.9 nM T20401 CD6Z0B 155566206 Ki = 4.4 nM T20401 COA9F8 155566222 Ki = 87200 nM T20401 CCW3L7 155566305 Ki = 837 nM T20401 CJQP47 155566378 Ki = 8.9 nM T20401 C5QAM3 155566668 Ki = 8.8 nM T20401 CBV30Y 155566701 Ki = 324.6 nM T20401 CA6JT2 155566730 Ki = 0.67 nM T20401 CI8U3W 155566755 Ki = 40.6 nM T20401 CA63FB 155566994 Ki = 9 nM T20401 CK80EL 155567119 Ki = 336.1 nM T20401 CC5A0I 155567282 Ki = 0.89 nM T20401 C4TZ8Q 155567475 Ki = 152.9 nM T20401 CK0M8P 155567487 Ki = 78.7 nM T20401 CL1N9Y 155567612 Ki > 100000 nM T20401 C1MHV5 155567738 Ki = 388.5 nM T20401 C29EYS 155567759 Ki = 790.6 nM T20401 CJ2YC4 155567804 Ki = 0.75 nM T20401 C9DOG1 155567981 Ki = 361.3 nM T20401 CZP30I 155567991 Ki = 8.5 nM T20401 CCX06Y 155568045 Ki = 1.2 nM T20401 CN5OF0 155568108 Ki = 5.6 nM T20401 CG8QF2 155568247 IC50 = 1500 nM T20401 C2ZRJ3 155568270 Ki = 52.4 nM T20401 CG82MB 155568274 Ki = 88.9 nM T20401 CDB8T4 155568445 Ki = 0.6 nM T20401 C94QKZ 155568447 Ki = 8.1 nM T20401 C52NQU 155568453 Ki = 4.1 nM T20401 C35XQY 155568474 Ki > 10000 nM T20401 C6KR4H 155568759 Ki = 466.3 nM T20401 CQM46K 155568895 IC50 = 2130 nM T20401 CH5VU6 155568899 Ki = 8.3 nM T20401 C1C2GI 155569076 Ki = 1.5 nM T20401 C83MGT 155569151 Ki = 7.5 nM T20401 CAUR85 155569555 Ki = 2200 nM T20401 C1A7IN 155569676 Ki = 5 nM T20401 D00BMI 25154729 Ki = 970 nM T20401 D00CIW 15295 Ki = 99 nM T20401 D00FGB 11414131 Ki = 1 nM T20401 D00GVA 44520904 Ki = 74 nM T20401 D00IAE 11974340 Ki = 45 nM T20401 D00IKQ 46703766 Ki = 93.8 nM T20401 D00IUB 13019 Ki = 108 nM T20401 D00LFX 20718630 Ki = 13 nM T20401 D00NUK 2837872 Ki = 64 nM T20401 D00OBI 9859866 Ki = 25 nM T20401 D00RDE 44246261 Ki = 93 nM T20401 D00RJT 943 Ki = 35000000 nM T20401 D00RNZ 910172 Ki = 50300 nM T20401 D00SXO 2793709 Ki > 10000 nM T20401 D00TRF 44423683 Ki = 94000 nM T20401 D00XIB 11680415 Ki = 19 nM T20401 D00XJA 711717 Ki = 13400 nM T20401 D00YEF 148885 Ki = 24.5 nM T20401 D01BUB 94952 Ki = 870000 nM T20401 D01CXM 52949265 Ki > 100000 nM T20401 D01EEM 462919 Ki = 16 nM T20401 D01FOK 52949288 Ki > 100000 nM T20401 D01GNQ 44395086 Ki = 49200000 nM T20401 D01ISX 670786 Ki = 53 nM T20401 D01JTI 11687831 Ki = 565 nM T20401 D01KKU 5281894 Ki = 2240 nM T20401 D01KOO 13654029 Ki = 1020 nM T20401 D01OTW 46703932 Ki = 91.1 nM T20401 D01STY 9861037 Ki = 70 nM T20401 D01UDU 11287480 Ki = 76 nM T20401 D01UYI 5281607 Ki = 4310 nM T20401 D01XFH 11851424 Ki = 47 nM T20401 D01YHK 10932611 Ki = 51 nM T20401 D02BMV 46907399 Ki = 108 nM T20401 D02DBP 5054 Ki = 7700 nM T20401 D02DCD 45483280 Ki = 184.5 nM T20401 D02JEZ 5281426 Ki > 10000 nM T20401 D02KDH 11160546 Ki = 264 nM T20401 D02MAK 5705744 Ki > 100000 nM T20401 D02NQK 46703924 Ki = 84.5 nM T20401 D02QGI 273 Ki = 11000 nM T20401 D03APP 4386 Ki = 38 nM T20401 D03DAM 2725651 Ki = 230 nM T20401 D03KRB 45028567 Ki = 65 nM T20401 D03LHJ 52946829 Ki > 100000 nM T20401 D03MJM 45273020 IC50 = 632000 nM T20401 D03NBX 637308 Ki > 50000 nM T20401 D03VUQ 404202 Ki = 11.1 nM T20401 D03ZMQ 323 Ki = 9200 nM T20401 D04BKU 148886 Ki = 9.7 nM T20401 D04CVC 4687472 Ki = 60 nM T20401 D04GDW 16098578 IC50 = 526 nM T20401 D04HQK 394898 Ki = 2 nM T20401 D04HRS 404195 Ki = 665 nM T20401 D04JIN 44405179 Ki = 112 nM T20401 D04LNI 75490 Ki = 4050 nM T20401 D04MAM 11356944 IC50 = 130 nM T20401 D04NSN 169682 Ki = 36.8 nM T20401 D04POB 8482 Ki = 246 nM T20401 D04PSK 44571848 Ki = 920 nM T20401 D04RCR 11041016 Ki = 18100 nM T20401 D04SNH 46933593 Ki = 80 nM T20401 D04VSP 46703768 Ki = 76.7 nM T20401 D05BMD 44423684 Ki = 4800 nM T20401 D05DIH 45483180 Ki = 158.4 nM T20401 D05EBZ 46703769 Ki = 94.5 nM T20401 D05ETN 46703923 Ki = 80.4 nM T20401 D05FMD 9447 IC50 = 720 nM T20401 D05FNN 100606 Ki = 8 nM T20401 D05JAJ 45028568 Ki = 105 nM T20401 D05KTE 6224 Ki = 2160000 nM T20401 D05NFU 4100860 Ki = 8700 nM T20401 D05PRS 296284 IC50 = 3600 nM T20401 D05QEK 44395692 Ki = 0.9 nM T20401 D05QOR 5280460 Ki > 100000 nM T20401 D05QUG 45485279 Ki = 40200 nM T20401 D05RAB 45028895 Ki = 77 nM T20401 D05TLB 11117301 Ki = 2.6 nM T20401 D05VUA 850202 Ki > 100000 nM T20401 D05VVC 44315786 Ki > 10000 nM T20401 D05WQF 637540 Ki = 9200 nM T20401 D05XZM 10081162 Ki = 8 nM T20401 D06ALC 6441498 Ki > 10000 nM T20401 D06DYP 234562 Ki = 62200 nM T20401 D06GPL 44405177 Ki = 348 nM T20401 D06IOI 901953 Ki = 9.9 nM T20401 D06IYU 15569631 Ki = 12 nM T20401 D06JVR 44571849 Ki = 870 nM T20401 D06KTD 2490720 Ki = 338 nM T20401 D06LVE 22784 IC50 = 400 nM T20401 D06MZK 31405 Ki = 510 nM T20401 D06NDR 44423687 Ki = 6100 nM T20401 D06ORV 65389 Ki = 17900 nM T20401 D06SME 46871781 IC50 = 6030 nM T20401 D06SZG 44315523 Ki > 10000 nM T20401 D06TPF 1057 Ki = 540 nM T20401 D06WZG 50925425 Ki > 100000 nM T20401 D06XNT 4119643 Ki = 54 nM T20401 D06XVV 64048 Ki > 500000 nM T20401 D06ZMH 2812287 Ki = 150 nM T20401 D06ZOM 15569045 Ki > 10000 nM T20401 D07AGM 14612854 Ki = 81.28 nM T20401 D07AUN 969280 Ki = 141.5 nM T20401 D07CBA 44391592 Ki = 563 nM T20401 D07CQI 42546 Ki = 420 nM T20401 D07CYN 20347846 Ki = 28 nM T20401 D07IHP 44391650 Ki = 9.4 nM T20401 D07IRQ 7478 Ki = 8030 nM T20401 D07JYF 13393427 IC50 = 250 nM T20401 D07LYW 11537386 Ki = 0.9 nM T20401 D07MQB 10903168 Ki = 29 nM T20401 D07MTM 403 Ki = 752000 nM T20401 D07OMY 44574267 Ki = 31 nM T20401 D07PNA 11660633 Ki = 128 nM T20401 D07PZQ 68841 Ki = 420000 nM T20401 D07QIU 625902 Ki = 464 nM T20401 D07QJJ 289 Ki = 9900 nM T20401 D07SIA 78318 Ki = 645 nM T20401 D07TAJ 914298 Ki = 24900 nM T20401 D07UCQ 23680200 Ki = 58300 nM T20401 D07VXX 16721024 Ki = 267000 nM T20401 D07YDN 5281654 Ki = 440 nM T20401 D07YSQ 10385283 Ki = 5 nM T20401 D07ZHE 67138 IC50 = 410 nM T20401 D07ZXR 44391576 Ki = 84.2 nM T20401 D08AIJ 440735 Ki > 10000 nM T20401 D08AOA 11543564 Ki = 10 nM T20401 D08BFU 5282102 Ki = 168 nM T20401 D08JCC 46703770 Ki = 94.4 nM T20401 D08JNO 52943193 Ki > 100000 nM T20401 D08ORD 45483187 Ki = 8.6 nM T20401 D08TCV 5988 Ki > 20000 nM T20401 D08XQI 9395 IC50 = 59 nM T20401 D09CSP 3161908 Ki = 495 nM T20401 D09CXX 16122590 Ki = 566 nM T20401 D09FQL 16756780 Ki = 11700 nM T20401 D09JHA 33558 Ki = 1500000 nM T20401 D09JPC 16402 Ki = 34400 nM T20401 D09LUD 4229592 Ki = 75 nM T20401 D09LWR 3433937 Ki = 67 nM T20401 D09OSN 151253 Ki = 4500 nM T20401 D09PUF 9842809 IC50 = 376 nM T20401 D09PWX 8739 Ki = 33 nM T20401 D09QHC 7370 Ki = 305 nM T20401 D09SFY 136123546 Ki = 236 nM T20401 D09TES 44395768 Ki = 65 nM T20401 D09TKG 25044690 Ki = 133 nM T20401 D09UQM 97463 Ki = 310 nM T20401 D09USO 5277466 IC50 = 9371 nM T20401 D09WSJ 19772348 Ki = 0.7 nM T20401 D09WVV 8111 Ki = 118000 nM T20401 D09ZUN 10269 Ki = 420 nM T20401 D0A0RT 11602828 Ki = 1870 nM T20401 D0A0YX 5143 Ki = 5180 nM T20401 D0A1CM 5281855 Ki = 2180 nM T20401 D0A3JR 3051968 Ki = 58 nM T20401 D0A4HS 201262 Ki = 7900 nM T20401 D0A4TC 446504 Ki = 8600 nM T20401 D0A5XB 11264735 IC50 = 280 nM T20401 D0A6HS 6852129 IC50 = 4 nM T20401 D0A8HW 44395685 Ki = 7.5 nM T20401 D0AU0M 637542 Ki = 980 nM T20401 D0B0SD 104745 Ki = 960000 nM T20401 D0B4IN 375084 Ki = 4975 nM T20401 D0B5GC 11349 Ki = 9200 nM T20401 D0BD0K 405487 Ki = 106 nM T20401 D0BR1D 13443185 IC50 = 2800 nM T20401 D0C3SL 67185 Ki = 290 nM T20401 D0C4QB 44395769 Ki = 84 nM T20401 D0C6ED 44564283 Ki = 643 nM T20401 D0C7LR 313 Ki = 200000000 nM T20401 D0C7WG 135932620 Ki = 106 nM T20401 D0C8ZY 2734375 Ki = 6000 nM T20401 D0C9ZY 11804953 Ki = 1250 nM T20401 D0CM3O 446142 Ki = 580000 nM T20401 D0D0BO 180598 Ki = 87 nM T20401 D0D1HC 46871782 IC50 = 7970 nM T20401 D0D2JA 2734377 Ki = 11500 nM T20401 D0D4OV 20043772 Ki = 14.6 nM T20401 D0D5XC 101753 Ki = 8800 nM T20401 D0D6UR 12394434 Ki = 7800 nM T20401 D0DY9U 23645365 Ki = 27 nM T20401 D0E0RW 69894 Ki > 100000 nM T20401 D0E3VJ 25154731 Ki = 1130 nM T20401 D0E8CC 18794 Ki = 9 nM T20401 D0EH0S 52943164 Ki > 100000 nM T20401 D0EJ9B 66827 Ki = 23.1 nM T20401 D0EX9Q 10881548 Ki = 115 nM T20401 D0EY2F 52949920 Ki > 100000 nM T20401 D0F3UR 690836 Ki = 469 nM T20401 D0F4ZW 46865217 IC50 = 122 nM T20401 D0F7KC 14116752 Ki > 100000 nM T20401 D0F7QZ 5702628 Ki = 534000 nM T20401 D0F7SO 94464 Ki = 125 nM T20401 D0FD8G 6011033 Ki = 373000 nM T20401 D0FU0K 23354226 Ki > 10000 nM T20401 D0G0BJ 51000408 Ki > 50000 nM T20401 D0G0FJ 11206245 Ki = 78 nM T20401 D0G0OP 44423685 Ki = 4700 nM T20401 D0G0ZI 403788 Ki = 8180 nM T20401 D0G3BI 25090 Ki = 9100 nM T20401 D0G3TK 5280863 Ki = 9525.7 nM T20401 D0G6OW 23675285 Ki = 6000 nM T20401 D0G9NE 11659798 Ki = 32 nM T20401 D0GI2R 11572651 IC50 = 8400 nM T20401 D0GQ9A 44593649 Ki = 49200000 nM T20401 D0H3NS 10752 Ki > 500000 nM T20401 D0H4CF 44246267 Ki = 88 nM T20401 D0HN0R 11623958 Ki = 118 nM T20401 D0I1XT 45483206 Ki = 38.5 nM T20401 D0I5YQ 44405178 Ki = 113 nM T20401 D0I8DW 612414 Ki = 13 nM T20401 D0IB3K 5320686 Ki > 10000 nM T20401 D0IU3X 44405186 Ki = 98 nM T20401 D0J1PZ 2723687 Ki = 8800 nM T20401 D0J2AE 7377 Ki = 240 nM T20401 D0J3SP 11718391 Ki = 6.7 nM T20401 D0J7GU 46703929 Ki = 40.1 nM T20401 D0J7KJ 52940758 Ki > 100000 nM T20401 D0K1FG 5411574 Ki > 100000 nM T20401 D0K3LN 3510137 Ki = 227 nM T20401 D0K4IH 687887 Ki = 123.2 nM T20401 D0K5NQ 10421755 Ki = 7 nM T20401 D0KB6T 721954 Ki = 37 nM T20401 D0KZ2D 11638641 Ki = 1.2 nM T20401 D0L1AV 45273021 IC50 = 181000 nM T20401 D0L2GD 60167587 Ki = 560000 nM T20401 D0L4FM 11030308 Ki = 1.3 nM T20401 D0L5TZ 20195365 Ki = 19200 nM T20401 D0L5XK 92249 Ki > 200000 nM T20401 D0L8ZG 79799 Ki = 10800 nM T20401 D0LC0F 96876 Ki = 52 nM T20401 D0LJ5P 44457221 Ki = 5.1 nM T20401 D0LM8L 11623927 IC50 = 3700 nM T20401 D0LU4S 156219 Ki = 38600 nM T20401 D0M3PO 69561 Ki = 62 nM T20401 D0M4EV 18975977 Ki = 16 nM T20401 D0M5MI 4306515 IC50 > 100000 nM T20401 D0M6RM 7365 Ki = 49.2 nM T20401 D0M7DE 11521450 IC50 = 7100 nM T20401 D0M7VN 44392435 Ki = 300 nM T20401 D0M8UY 72139 IC50 = 1770 nM T20401 D0M9IQ 23665438 Ki = 63600 nM T20401 D0N0JL 1023 Ki = 48500000 nM T20401 D0N1AW 45485270 Ki = 18500 nM T20401 D0N5KX 44391625 Ki = 643 nM T20401 D0N7WP 44520903 Ki = 69 nM T20401 D0N8LR 847760 Ki = 232 nM T20401 D0N8VZ 11583423 Ki = 232 nM T20401 D0NN3Q 78105 IC50 = 80 nM T20401 D0NS0E 220188 Ki > 10000 nM T20401 D0O0UE 729977 Ki = 9 nM T20401 D0O1QT 93505 Ki = 9 nM T20401 D0O4KL 11640067 Ki = 490 nM T20401 D0O6ZD 14101447 Ki > 100000 nM T20401 D0O8WV 11536481 Ki = 46 nM T20401 D0O9VU 44520901 Ki = 61 nM T20401 D0OC4B 5357479 Ki > 10000 nM T20401 D0OI1H 72894 Ki = 295 nM T20401 D0OT5L 1631814 Ki = 29000 nM T20401 D0P6AM 3526523 Ki = 40 nM T20401 D0PA5L 44380941 Ki = 32 nM T20401 D0Q0EK 318174 Ki = 124 nM T20401 D0Q0XO 4258082 Ki = 214 nM T20401 D0Q1EI 3084733 Ki = 73 nM T20401 D0Q2XB 75928 Ki = 339790 nM T20401 D0Q5VB 46704078 Ki = 87.2 nM T20401 D0Q7DJ 10742 Ki = 3190 nM T20401 D0R4KQ 46704077 Ki = 140 nM T20401 D0R4WJ 16129778 Ki = 32800 nM T20401 D0R6JK 2306645 Ki = 200.5 nM T20401 D0R7QY 127676 IC50 = 9 nM T20401 D0RB0D 44268050 Ki = 49500 nM T20401 D0RK7J 235259 Ki = 133 nM T20401 D0S0RK 10680 Ki = 8710 nM T20401 D0S1OY 10946908 Ki = 96 nM T20401 D0S2II 308405 Ki = 21.4 nM T20401 D0S3RZ 9954405 Ki = 5 nM T20401 D0S4NO 25154730 Ki = 950 nM T20401 D0S9YX 5280373 Ki > 10000 nM T20401 D0SF3B 11529486 Ki = 7.5 nM T20401 D0SV6C 8625 Ki = 13000 nM T20401 D0SY2M 5281708 Ki > 10000 nM T20401 D0T0YI 378 IC50 = 63 nM T20401 D0T2VH 44571846 Ki = 900 nM T20401 D0T2YZ 3253857 Ki = 258 nM T20401 D0T3NP 7456 Ki = 3400 nM T20401 D0T6VB 521293 Ki = 30000 nM T20401 D0T8SN 12033284 Ki = 11 nM T20401 D0T9BB 52950111 Ki > 100000 nM T20401 D0TY8X 31036 Ki = 12 nM T20401 D0U0QW 45483186 Ki = 160 nM T20401 D0U1AN 521359 Ki = 185 nM T20401 D0U4BB 10748 Ki > 500000 nM T20401 D0UM1I 12554666 Ki = 85.6 nM T20401 D0UN0E 12195854 Ki = 156 nM T20401 D0V0FY 52946831 Ki > 100000 nM T20401 D0V5OW 46907400 Ki = 131 nM T20401 D0V9EN 689043 Ki = 1610 nM T20401 D0VD7H 84724 Ki = 60 nM T20401 D0W1AW 4234241 Ki = 6.6 nM T20401 D0W1OR 7424 Ki = 510 nM T20401 D0W2XO 6364608 Ki = 989000 nM T20401 D0W9VC 670143 Ki = 50 nM T20401 D0X0PO 20043771 Ki = 8.3 nM T20401 D0X0RE 6019835 Ki = 617000 nM T20401 D0X1MY 2723847 Ki = 9200 nM T20401 D0X5HL 15107 Ki = 103000 nM T20401 D0X6IE 4422372 Ki = 30 nM T20401 D0X9LJ 788811 Ki = 100 nM T20401 D0XK7G 10445302 Ki = 32 nM T20401 D0XL5K 67944 Ki = 30 nM T20401 D0Y1XM 44423686 Ki = 7800 nM T20401 D0Y3TZ 370 Ki = 2250 nM T20401 D0Y7HG 5281616 Ki > 10000 nM T20401 D0YD9F 822774 Ki = 49 nM T20401 D0YU8J 1502014 Ki = 110 nM T20401 D0YZ5G 5281416 Ki > 10000 nM T20401 D0Z1CL 79599 Ki = 7000 nM T20401 D0Z1HY 67136 Ki = 75 nM T20401 D0Z5GE 44520902 Ki = 395 nM T20401 D0Z6TM 3558590 Ki = 47 nM T20401 D0ZC3W 6269 Ki = 320 nM T35940 D04XVN 11707110 IC50 = 0.7 nM T35940 D0K8KX 5280343 IC50 > 10000 nM T35940 D0OB0F 5328940 IC50 = 1 nM T35940 D0T5DP 10127622 IC50 = 14 nM T35940 D01CNB 10172827 IC50 = 50 nM T35940 D01IED 11719003 IC50 > 10000 nM T35940 D02UFQ 11620908 IC50 = 1100 nM T35940 D03CHM 44187362 IC50 = 1.81 nM T35940 D07DTV 11338033 IC50 > 10000 nM T35940 D0B9BU 6918454 IC50 = 2 nM T35940 D0E3TC 44259 IC50 = 2.5 nM T35940 D0I3RD 24963252 IC50 = 3.2 nM T35940 D0K0YC 9826528 IC50 = 7 nM T35940 D0M6BD 16719221 IC50 = 160 nM T35940 D0O2FN 16222096 IC50 = 0.9 nM T35940 D0Q4IX 71727581 IC50 > 10000 nM T35940 D0VF6E 1401 IC50 > 50000 nM T35940 D03BNU 59604787 IC50 > 3500 nM T35940 D02GEJ 5326976 IC50 = 10500 nM T35940 C8KED5 4713 IC50 = 2000 nM T35940 C5HUE3 64981 IC50 = 1 nM T35940 C4MNG8 445840 IC50 > 10000 nM T35940 CJ4QI8 885402 IC50 = 200 nM T35940 CQ7PL4 1235170 IC50 > 20000 nM T35940 C4WFP1 1587957 IC50 = 12300 nM T35940 C9EUD2 1839691 IC50 = 8500 nM T35940 C1SVD2 2132479 IC50 = 9000 nM T35940 CKLG52 2726558 IC50 = 410 nM T35940 C2PB6W 2726567 IC50 > 5000 nM T35940 C5GYO1 2730801 IC50 = 300 nM T35940 CAXR02 3338590 IC50 > 5000 nM T35940 CK27AT 3694944 IC50 = 18100 nM T35940 C8IAR2 5281657 IC50 > 100000 nM T35940 CI68PW 5283685 IC50 > 100000 nM T35940 CXK0S6 5283727 IC50 = 48900 nM T35940 C94GRU 5330453 IC50 = 280 nM T35940 C4G9WR 9547398 IC50 > 100000 nM T35940 C76CUP 9547698 IC50 > 100000 nM T35940 CSNH60 9803891 IC50 = 2 nM T35940 CNA9K2 9806897 IC50 = 1.1 nM T35940 CK2J3G 9863776 IC50 = 2.9 nM T35940 CW8V0K 9864418 IC50 > 50000 nM T35940 C18HKQ 9885748 IC50 = 12800 nM T35940 CHF7G5 9890746 IC50 > 30000 nM T35940 C2Y3WG 9907612 IC50 = 4900 nM T35940 C3EUB4 9911005 IC50 > 30000 nM T35940 C07VNB 9930243 IC50 = 6 nM T35940 CJO47T 9948405 IC50 > 10000 nM T35940 CH57ND 9951825 IC50 = 2600 nM T35940 C3I5HT 9978125 IC50 = 6.2 nM T35940 C37GXK 9983303 IC50 = 40 nM T35940 CV8I5X 9999342 IC50 > 10000 nM T35940 CR8DA1 10024683 IC50 > 100000 nM T35940 CLA93G 10047202 IC50 > 100000 nM T35940 C3LCH5 10047545 IC50 > 100000 nM T35940 C2C1BP 10089048 IC50 = 20000 nM T35940 C0Y5PD 10118314 IC50 = 650 nM T35940 CC5Q3G 10135899 IC50 = 7.7 nM T35940 CH4W9D 10139826 IC50 = 2 nM T35940 C3NW6G 10164464 IC50 = 72 nM T35940 CNJ91A 10185285 IC50 = 14 nM T35940 CJ09AO 10185838 IC50 = 29 nM T35940 C5LUV3 10206034 IC50 = 10 nM T35940 CD3OV6 10206158 IC50 = 0.6 nM T35940 C9XBD5 10225656 IC50 = 10 nM T35940 CMN70R 10228676 IC50 = 20 nM T35940 C5TQ7X 10247543 IC50 > 10000 nM T35940 C1AKH9 10303277 IC50 = 8 nM T35940 CN23SU 10324074 IC50 = 7 nM T35940 CK82OA 10345719 IC50 = 25 nM T35940 C4CP7K 10423452 IC50 > 100000 nM T35940 C95LYF 10457505 IC50 > 30000 nM T35940 CHM9I6 10461359 IC50 = 2 nM T35940 C2WQ8M 10473563 IC50 > 10000 nM T35940 CRX6F0 10479082 IC50 = 200 nM T35940 C83QWV 10714343 IC50 > 100000 nM T35940 CJ4P5T 10905857 IC50 > 30000 nM T35940 C3ZE1P 11064594 IC50 = 2500 nM T35940 CV2O1Z 11165133 IC50 = 43 nM T35940 C82QDW 11188772 IC50 = 30 nM T35940 C8G5WP 11210533 IC50 > 30000 nM T35940 C2W5RC 11235063 IC50 > 25000 nM T35940 C0QA8R 11236142 IC50 = 124 nM T35940 C73WRC 11281076 IC50 = 33 nM T35940 CB6OM9 11384425 IC50 = 18 nM T35940 C13CZV 11395411 IC50 = 82 nM T35940 C0HEN9 11418932 IC50 = 6.8 nM T35940 C0APW4 11422034 IC50 > 10000 nM T35940 C58PRM 11439749 IC50 = 14 nM T35940 CDQ31C 11485916 IC50 = 105 nM T35940 CT9V3D 11496376 IC50 = 630 nM T35940 C0QG4W 11523601 IC50 = 118 nM T35940 CRP2U5 11526671 IC50 = 23 nM T35940 C7HMO6 11526786 IC50 > 10000 nM T35940 CO9KP5 11583459 IC50 > 10000 nM T35940 C0WJX2 11603973 IC50 = 2200 nM T35940 C2OMY7 11611241 IC50 = 39 nM T35940 C2HY5O 11613319 EC50 = 49 nM T35940 CGJ2A0 11617424 IC50 = 30 nM T35940 CK34LS 11632737 IC50 > 5000 nM T35940 CWIH62 11633097 IC50 = 9.3 nM T35940 CP4T3N 11669238 IC50 = 45 nM T35940 CJ9KN7 11683817 IC50 > 10000 nM T35940 CZFH19 11689297 IC50 = 15 nM T35940 CSJ69K 11690375 IC50 = 40 nM T35940 CU0E8O 11690457 Ki > 1000 nM T35940 CB0AP2 11705863 Ki > 10000 nM T35940 C9P0VD 11729539 IC50 > 30000 nM T35940 CPN42M 11755998 IC50 = 2.7 nM T35940 CO3QF7 15951576 IC50 = 1200 nM T35940 C7RUN8 15984125 IC50 = 38 nM T35940 C9TU1O 16046126 IC50 > 1000 nM T35940 CZHJ34 16058637 IC50 = 6800 nM T35940 CKV4G1 16079040 IC50 = 1100 nM T35940 CKX2L7 16085320 IC50 = 960 nM T35940 C4V0CW 16126717 IC50 = 28 nM T35940 C5VPH9 16129448 IC50 = 139 nM T35940 C3KB2P 16221892 IC50 = 7.6 nM T35940 CY8B2U 16221995 IC50 = 5.1 nM T35940 C5PXQ4 16222191 IC50 = 6.6 nM T35940 CD3SV4 16222192 IC50 = 5.2 nM T35940 CC5NK6 16222193 IC50 = 16 nM T35940 CX5H2Q 16222302 IC50 = 1708 nM T35940 CR0HT5 16222819 IC50 = 1.8 nM T35940 C6CHI8 16222917 IC50 = 220 nM T35940 CVYD02 16222921 IC50 = 7.2 nM T35940 CF5PJ6 16223027 IC50 = 4.8 nM T35940 C4PVA3 16223325 IC50 = 44 nM T35940 C1AN2Q 16223412 IC50 = 535 nM T35940 C0A5HN 16223413 IC50 = 27 nM T35940 CA80DB 16223418 IC50 = 82 nM T35940 CE2U1Y 16655058 IC50 = 800 nM T35940 C2IF3P 16678352 IC50 = 960 nM T35940 C3IO1C 16679060 IC50 > 10000 nM T35940 CG05KJ 16720763 IC50 = 25 nM T35940 C5FEX0 16727871 IC50 > 5000 nM T35940 CQ79FH 16727872 IC50 > 5000 nM T35940 CP81ZK 16727873 IC50 > 5000 nM T35940 CJ9QN3 16727876 IC50 > 5000 nM T35940 CA6W3J 16727880 IC50 > 5000 nM T35940 C3J4GL 16727881 IC50 = 650 nM T35940 C81MEA 16727889 IC50 = 250 nM T35940 C7UT6L 16727891 IC50 > 5000 nM T35940 CC2XV5 16727892 IC50 > 5000 nM T35940 CN6A7C 16727895 IC50 > 5000 nM T35940 CT0FB2 16727911 IC50 > 5000 nM T35940 C6IM0U 16727912 IC50 > 5000 nM T35940 CO7C9M 16727913 IC50 > 5000 nM T35940 CEF64U 17599247 IC50 = 23100 nM T35940 CAV35B 17903650 IC50 = 26 nM T35940 CNY91P 20791410 IC50 = 33 nM T35940 C1GH5L 20791412 IC50 = 24 nM T35940 CH8A1O 20791416 IC50 = 29 nM T35940 C8KIW5 20791505 IC50 = 48 nM T35940 CZFE08 20791507 IC50 = 76 nM T35940 CKV3A0 20791510 IC50 = 58 nM T35940 C8UTF2 20791535 IC50 = 14 nM T35940 CU36BS 20791561 IC50 > 25000 nM T35940 CP5O8N 20791586 IC50 = 23 nM T35940 C3OTW0 20791598 IC50 = 566 nM T35940 C2WB5M 20791599 IC50 = 331 nM T35940 CKI91V 20791601 IC50 = 203 nM T35940 CV5WM3 20791602 IC50 = 191 nM T35940 C5X3IH 20791605 IC50 = 2650 nM T35940 CR51GI 20791606 IC50 = 5420 nM T35940 CO97JA 20791607 IC50 > 25000 nM T35940 C5EMT7 20791608 IC50 > 25000 nM T35940 CJPS16 20791615 IC50 = 642 nM T35940 CPD4J0 20791616 IC50 = 2320 nM T35940 CB6Z5Q 20791617 IC50 = 1110 nM T35940 CRK28W 20791618 IC50 > 25000 nM T35940 C8BT9L 20791619 IC50 = 68 nM T35940 C15NJF 20791626 IC50 > 25000 nM T35940 CN4W6G 20791639 IC50 = 23 nM T35940 C14YFA 21024387 IC50 = 96 nM T35940 CEQ2L7 21024393 IC50 = 10000 nM T35940 CKPC54 21025113 IC50 = 94 nM T35940 CR8H4Y 21110084 IC50 = 39400 nM T35940 C92GDY 21704772 IC50 = 4.2 nM T35940 CQ7BT0 21704776 IC50 = 33 nM T35940 CZJT36 21704852 IC50 = 5 nM T35940 CO2C7D 21704856 IC50 = 20 nM T35940 CT9N7Z 21808053 IC50 > 5000 nM T35940 CULN54 22025663 IC50 = 19.5 nM T35940 C7X3LY 22179466 IC50 = 147 nM T35940 C69UHM 22179477 IC50 = 36 nM T35940 CJN17H 22179480 IC50 = 6130 nM T35940 C83WSJ 22179488 IC50 = 190 nM T35940 CE35RW 22179532 IC50 = 241 nM T35940 C3CB0X 22179547 IC50 > 25000 nM T35940 CIBU26 22179588 IC50 = 42 nM T35940 CQ2WV5 22179590 IC50 = 14600 nM T35940 C4AKZ1 22179615 IC50 > 25000 nM T35940 CO1D8J 22179618 IC50 = 521 nM T35940 CMKR54 22179638 IC50 = 361 nM T35940 CL9RS7 22179671 IC50 = 181 nM T35940 CI68XT 22179674 IC50 = 18 nM T35940 CY47CN 22179680 IC50 = 168 nM T35940 C2DV7M 22179683 IC50 > 25000 nM T35940 CC6HS9 22179713 IC50 = 397 nM T35940 CXH2L0 22179728 IC50 = 87 nM T35940 COM5D6 22255964 IC50 = 500 nM T35940 CUSD96 22255970 IC50 > 5000 nM T35940 CKO7I9 22255979 IC50 > 5000 nM T35940 C51FVK 22255982 IC50 > 5000 nM T35940 CB13LM 22255988 IC50 > 5000 nM T35940 C8F4NU 22271692 IC50 = 26 nM T35940 CQMO93 22466681 IC50 = 280 nM T35940 CZX61A 22466740 IC50 = 100 nM T35940 C9I8EY 22473189 IC50 = 386 nM T35940 CQRV31 22743091 IC50 = 8 nM T35940 CYUX63 22743123 IC50 = 17 nM T35940 CWQC81 22743127 IC50 = 8 nM T35940 CG6D4M 23647319 IC50 > 10000 nM T35940 CY8Z7X 23647330 IC50 > 10000 nM T35940 C4XD8H 23647348 IC50 > 10000 nM T35940 CN20YH 24743899 EC50 = 6.3 nM T35940 C6JCE7 24753323 IC50 = 28 nM T35940 C50GZI 24753409 IC50 = 53 nM T35940 CC4RZ6 24753410 IC50 = 230 nM T35940 CB3D1Y 24753411 IC50 = 110 nM T35940 C6JF2R 24753412 IC50 = 9 nM T35940 CWX89I 24753603 IC50 = 60 nM T35940 C4CY3V 24753607 IC50 = 110 nM T35940 CFN72M 24753694 IC50 = 64 nM T35940 CQJ2D3 24753784 IC50 = 38 nM T35940 CP1E4R 24753786 IC50 = 99 nM T35940 CA3I4T 24753787 IC50 = 7 nM T35940 CW36DL 24753877 IC50 = 66 nM T35940 COAY09 24753878 IC50 = 97 nM T35940 C9H7EZ 24753971 IC50 = 59 nM T35940 C6CT7I 24753973 IC50 = 26 nM T35940 CS98MR 24754053 IC50 = 46 nM T35940 C9Q3DE 24754054 IC50 = 47 nM T35940 CRJ9G6 24754132 IC50 = 36 nM T35940 CBD59Z 24754133 IC50 = 65 nM T35940 CKV76A 24754134 IC50 = 58 nM T35940 CM8HY9 24754207 IC50 = 4200 nM T35940 C7YG1N 24759534 IC50 = 7200 nM T35940 CM9ED1 24784164 IC50 = 18 nM T35940 C9PA0M 24807809 IC50 > 10000 nM T35940 C61KPI 24856363 IC50 > 50000 nM T35940 C2HEA1 24963248 IC50 = 4.8 nM T35940 CNS0P4 24963250 IC50 = 16 nM T35940 C2Z1GV 24963251 IC50 = 3.2 nM T35940 CF57BL 24963596 IC50 = 8.6 nM T35940 C2F6VC 24965727 IC50 = 26 nM T35940 C9MXU6 24965728 IC50 = 9.8 nM T35940 CQ5K9J 24965731 IC50 = 8.3 nM T35940 CG6PX7 24966075 IC50 = 3.8 nM T35940 CC1AS8 24966426 IC50 = 5 nM T35940 CDJZ34 24966428 IC50 = 4 nM T35940 CNR1E2 24967882 IC50 = 53 nM T35940 CQL29E 24967884 IC50 = 740 nM T35940 CNG6P3 24968231 IC50 = 4.9 nM T35940 CU7W2H 24968572 IC50 = 3.1 nM T35940 CF9UH3 24968575 IC50 = 3.3 nM T35940 C32AUW 25013308 IC50 = 12 nM T35940 C4QF6H 25101222 IC50 = 18000 nM T35940 CVHF49 25124153 IC50 = 17 nM T35940 C7JK8L 25124154 IC50 = 41 nM T35940 C3MUZ7 25124155 IC50 = 14 nM T35940 CI8W7P 25124156 IC50 = 32 nM T35940 CKLW04 25124159 IC50 = 52 nM T35940 C6OSI9 25124477 IC50 = 20 nM T35940 C4A0CP 25124478 IC50 = 76 nM T35940 CPC6N3 25124479 IC50 = 18 nM T35940 CF7BM9 25124819 IC50 = 8.9 nM T35940 CJ56ZC 25125162 IC50 = 54 nM T35940 CD4H7O 25125510 IC50 = 36 nM T35940 CRM79Y 25125842 IC50 = 11 nM T35940 CIUJ83 25167109 EC50 = 45 nM T35940 C6VNB2 25181191 IC50 = 19 nM T35940 CN5TH0 25186684 IC50 = 42 nM T35940 CYHE45 25186685 IC50 = 46 nM T35940 C1B0RC 25186686 IC50 = 20 nM T35940 C6MWK4 25186687 IC50 = 11 nM T35940 CST81A 25186959 IC50 = 32 nM T35940 CM4W6B 25186960 IC50 = 13 nM T35940 CKUI82 25186961 IC50 = 18 nM T35940 C65UMS 25186963 IC50 = 19 nM T35940 CWBI46 25187248 IC50 = 90 nM T35940 CS1F6O 25187538 IC50 = 7 nM T35940 CY07IE 25187543 IC50 = 30 nM T35940 C6DZN3 25187544 IC50 = 13 nM T35940 CZ87LE 25188088 IC50 = 19 nM T35940 C6FGQ1 25206346 IC50 = 1000 nM T35940 CRO09K 25211064 IC50 = 225 nM T35940 C8MBU1 25211459 IC50 = 1800 nM T35940 CF9O0S 25218754 IC50 = 9700 nM T35940 C4T7YX 25218756 IC50 = 13000 nM T35940 CM2GY7 25218822 IC50 = 3 nM T35940 CD80NJ 25218823 IC50 = 4 nM T35940 CT84WC 25218824 IC50 = 8 nM T35940 C6P0UZ 42606202 IC50 = 39 nM T35940 C7NZD9 42606204 IC50 = 25 nM T35940 CWN59K 42606205 IC50 = 94 nM T35940 CCO2Z0 42606316 IC50 = 57 nM T35940 C3ET7Q 42606317 IC50 = 38 nM T35940 CN72OJ 42606318 IC50 = 29 nM T35940 CHG6V0 42606319 IC50 = 109 nM T35940 CQG9O8 42606320 IC50 = 69 nM T35940 CU9E4P 42629114 IC50 > 10000 nM T35940 C48USC 44143344 IC50 = 15000 nM T35940 CM86PK 44143527 IC50 = 750 nM T35940 CC9SL5 44143531 IC50 = 660 nM T35940 CFP1N7 44143534 IC50 = 800 nM T35940 CEL61X 44229839 IC50 = 2100 nM T35940 CYE36B 44241613 IC50 > 40000 nM T35940 C6LG5T 44241614 IC50 > 40000 nM T35940 C90AGP 44279526 IC50 = 1100 nM T35940 C4EI5V 44279624 IC50 = 160 nM T35940 C6M1OS 44279650 IC50 = 3.6 nM T35940 CA0M5Q 44279651 IC50 = 210 nM T35940 CF1X7T 44279777 IC50 > 10000 nM T35940 CWEL07 44279868 IC50 = 550 nM T35940 CF87XG 44279881 IC50 = 3000 nM T35940 CD6CJ8 44279890 IC50 = 110 nM T35940 C5DBE9 44279911 IC50 = 99 nM T35940 C6J1OV 44279943 IC50 = 3300 nM T35940 C7H3PB 44279996 IC50 = 21 nM T35940 CZYS81 44283696 IC50 = 25 nM T35940 CD0EH5 44283728 IC50 = 140 nM T35940 C91FKW 44328166 IC50 = 35 nM T35940 C1PIV3 44328167 IC50 = 450 nM T35940 C68XOD 44328201 IC50 > 10000 nM T35940 CSU37A 44328224 IC50 > 10000 nM T35940 C1HX0W 44328247 IC50 = 68 nM T35940 CKE68U 44328248 IC50 > 10000 nM T35940 CM6B3A 44328249 IC50 = 185 nM T35940 CL5O9W 44328252 IC50 = 680 nM T35940 C65NIO 44328253 IC50 = 125 nM T35940 C0O4XE 44328572 IC50 = 1400 nM T35940 C2IS5Y 44328691 IC50 = 2100 nM T35940 CMW9F0 44328708 IC50 = 1900 nM T35940 CCP8J1 44328755 IC50 = 13500 nM T35940 CO0S3H 44333650 IC50 = 2 nM T35940 CJ16TV 44333771 IC50 = 28 nM T35940 CPC8D0 44333792 IC50 = 212 nM T35940 CH4NW2 44333813 IC50 = 1 nM T35940 C1Y2CA 44333834 IC50 = 2 nM T35940 CZ6OS0 44333854 IC50 = 9 nM T35940 CZ4VX0 44405504 IC50 = 800 nM T35940 CGNY76 44406797 IC50 = 6786 nM T35940 CLG76N 44406798 IC50 = 4496 nM T35940 C74NHO 44407254 IC50 = 3470 nM T35940 C08BQD 44407284 IC50 = 805 nM T35940 C0H6US 44413718 IC50 > 5000 nM T35940 CFYX93 44413976 IC50 = 740 nM T35940 CR6U0N 44413985 IC50 > 2000 nM T35940 CD20CK 44413990 IC50 > 2000 nM T35940 CE9G6B 44413993 IC50 > 5000 nM T35940 CI9AG7 44413998 IC50 = 620 nM T35940 CK6VP8 44414003 IC50 = 1390 nM T35940 CAY1K3 44414006 IC50 = 1440 nM T35940 C5CGN9 44414007 IC50 = 420 nM T35940 CU78XJ 44414009 IC50 = 500 nM T35940 C2O3RA 44414010 IC50 = 500 nM T35940 CCEI57 44414011 IC50 = 430 nM T35940 C8KHP9 44414015 IC50 = 1230 nM T35940 CW1OL5 44414016 IC50 = 350 nM T35940 CY9SE4 44414021 IC50 = 1450 nM T35940 C5Q7KO 44414022 IC50 > 5000 nM T35940 CN02UR 44414024 IC50 = 670 nM T35940 CYK80F 44414025 IC50 > 5000 nM T35940 CB2L1H 44414026 IC50 = 690 nM T35940 CER4G2 44414027 IC50 = 790 nM T35940 CHY41Q 44414028 IC50 = 410 nM T35940 CG60RC 44414372 IC50 = 62 nM T35940 C4TKO7 44414373 IC50 = 73 nM T35940 C7B9EF 44414374 IC50 = 42 nM T35940 CV15GH 44414396 IC50 = 44 nM T35940 CWLQ15 44414397 IC50 = 68 nM T35940 CUL41F 44414398 IC50 = 86 nM T35940 C1YFX2 44414420 IC50 = 220 nM T35940 CT37HL 44414550 IC50 = 510 nM T35940 CPQ83M 44414575 IC50 = 1440 nM T35940 CJAD46 44415333 IC50 > 5000 nM T35940 C06AMS 44415334 IC50 > 5000 nM T35940 C8IL7A 44415335 IC50 > 5000 nM T35940 C1VT7R 44417767 EC50 = 42 nM T35940 CI4JW0 44417768 EC50 = 130 nM T35940 CFN83L 44417769 EC50 = 100 nM T35940 CK73YC 44417770 IC50 = 45 nM T35940 C7TNE3 44417771 IC50 = 150 nM T35940 C6GJD3 44417772 EC50 = 1500 nM T35940 CA05IE 44417773 IC50 = 44 nM T35940 C2IX3Y 44417774 EC50 = 123 nM T35940 C82LKD 44417775 EC50 = 95 nM T35940 CLY7T6 44417776 EC50 = 350 nM T35940 C59VBJ 44417777 EC50 = 30 nM T35940 CN7QO0 44417778 EC50 = 130 nM T35940 CG76RQ 44417779 EC50 = 70 nM T35940 C7TZH3 44417780 EC50 = 88 nM T35940 CLGM87 44417781 EC50 = 330 nM T35940 CJ12MO 44417782 IC50 = 30 nM T35940 C4JG5U 44417783 EC50 = 260 nM T35940 CA8OE1 44417784 IC50 = 26 nM T35940 CAP9Q8 44417785 EC50 = 350 nM T35940 C3OGB8 44417786 EC50 > 10 nM T35940 C51HVW 44417787 EC50 = 100 nM T35940 CFI0Y5 44417788 IC50 = 20 nM T35940 C24RCB 44417789 EC50 > 10 nM T35940 C2YD6G 44417790 IC50 = 145 nM T35940 CZ0C9J 44417791 IC50 = 20 nM T35940 C68HYN 44417792 EC50 = 128 nM T35940 CU3IM9 44417793 IC50 = 85 nM T35940 CSQV34 44417794 EC50 = 37 nM T35940 CPE0C6 44417795 IC50 = 64 nM T35940 CKA7L6 44417796 EC50 = 150 nM T35940 CEJ97B 44417797 IC50 = 37 nM T35940 CV0QD3 44417798 IC50 = 27 nM T35940 CU1NE0 44417799 EC50 = 250 nM T35940 CY5DZ8 44417801 EC50 = 35 nM T35940 CO0L1N 44417802 EC50 = 284 nM T35940 CUK65S 44417804 EC50 = 118 nM T35940 C7PQM6 44417805 IC50 = 298 nM T35940 COBQ43 44417806 EC50 = 43 nM T35940 CAK81N 44417807 IC50 = 46 nM T35940 CE15NX 44417808 EC50 = 54 nM T35940 C8BJ4S 44417809 EC50 = 120 nM T35940 CL81HY 44417810 EC50 = 22 nM T35940 CQU84C 44417812 EC50 = 564 nM T35940 C3HF6D 44417813 EC50 = 694 nM T35940 CP9VZ5 44417814 EC50 = 65 nM T35940 CSH5V7 44417815 EC50 = 6190 nM T35940 C2I7LO 44468504 IC50 = 48 nM T35940 C2VMW6 44469046 IC50 = 182 nM T35940 CKF1D5 44469440 IC50 = 21 nM T35940 CTH3R7 44469586 IC50 = 539 nM T35940 C1TVZ8 44469864 IC50 = 32 nM T35940 C4V6YC 44470284 IC50 = 21 nM T35940 C1SZX9 44545708 EC50 = 0.2 nM T35940 C3VRO9 44557921 IC50 > 10000 nM T35940 CZI8O2 44580056 IC50 = 1500 nM T35940 C4YOF5 44580057 IC50 = 1900 nM T35940 CQL65I 44580058 IC50 = 7600 nM T35940 CV0WF3 44580059 IC50 = 1500 nM T35940 C7Q1VU 44580077 IC50 = 30 nM T35940 CM7DC1 44580107 IC50 = 48000 nM T35940 C5JMS7 44580231 IC50 = 14000 nM T35940 CK1VE7 44580420 IC50 = 400 nM T35940 CEKG17 44580755 IC50 = 21800 nM T35940 CX7E6T 44580756 IC50 = 2400 nM T35940 C5V3PQ 44580757 IC50 = 21200 nM T35940 CXNQ42 44580758 IC50 = 23000 nM T35940 CR9LU0 44580759 IC50 = 49000 nM T35940 C0L9DI 44588712 IC50 = 35 nM T35940 CW2K3V 44588713 IC50 = 36 nM T35940 CM1AR5 44588714 IC50 = 5 nM T35940 CG9CK2 44588732 IC50 = 59 nM T35940 C4IYE2 44588733 IC50 = 55 nM T35940 CNC6I3 44588734 IC50 = 52 nM T35940 CM3Y0O 44588735 IC50 = 26 nM T35940 C3SYC8 44588760 IC50 = 21 nM T35940 CUYD68 44588761 IC50 = 11 nM T35940 CD02AX 44588762 IC50 = 20 nM T35940 CV9ZW5 44588763 IC50 = 10 nM T35940 CZ7LX5 44588812 IC50 = 33 nM T35940 C67ULC 44588813 IC50 = 3 nM T35940 CH13YD 44588814 IC50 = 4 nM T35940 CSTB61 44588815 IC50 = 6 nM T35940 C5Z3LI 44591740 IC50 > 30000 nM T35940 C2DY3A 44603143 EC50 = 0.4 nM T35940 CW2K8V 44603144 EC50 = 3.4 nM T35940 CJ5CH4 44603148 EC50 = 1.3 nM T35940 CO7DT3 44603204 EC50 = 1.5 nM T35940 CMQ0T2 44603207 IC50 = 4546 nM T35940 C4MOE2 44603271 EC50 = 0.6 nM T35940 C87WRB 44603341 EC50 = 0.9 nM T35940 C87FEM 45270051 IC50 > 40000 nM T35940 CU53FK 45273505 IC50 > 40000 nM T35940 CO7Q2F 46186796 IC50 = 15 nM T35940 CBQ3P6 46195697 IC50 = 18 nM T35940 C4U2MA 46196215 IC50 = 36 nM T35940 CUA97D 46209401 IC50 = 3700 nM T35940 C1J6GR 46224908 IC50 > 10000 nM T35940 CZ20AF 49797945 IC50 = 220 nM T35940 C14NZO 49797965 IC50 = 72 nM T35940 C03FHV 49797966 IC50 = 11 nM T35940 CQ4J0V 49797967 IC50 = 20 nM T35940 C4O9ZB 49798006 IC50 = 29 nM T35940 CHSF07 49806372 IC50 > 1000 nM T35940 CB0S2P 49842666 IC50 = 22000 nM T35940 CAI20B 49842778 IC50 = 12000 nM T35940 CRA74I 49842779 IC50 = 17000 nM T35940 CQUS34 51347355 IC50 = 8.7 nM T35940 CEQN27 52936621 Ki > 1000 nM T35940 CM24LF 52938983 IC50 = 18.19 nM T35940 CF04QJ 53318508 IC50 = 5.9 nM T35940 CZY0J7 53323592 IC50 > 100000 nM T35940 C5TED6 53323815 IC50 = 4.6 nM T35940 CNPM14 53341082 IC50 > 3000 nM T35940 C8G4RK 54016394 IC50 = 300000 nM T35940 C9ZFS1 54764923 IC50 > 100000 nM T35940 CT4E8R 56832546 IC50 = 30000 nM T35940 C6O5WH 56951292 IC50 > 10000 nM T35940 CR0Q2N 57523121 IC50 > 10000 nM T35940 C6CUN1 57624898 IC50 = 69 nM T35940 CE23DS 57624909 IC50 = 21 nM T35940 C7F2XZ 57624940 IC50 = 43 nM T35940 CGU9R7 57624954 IC50 = 96 nM T35940 CX8W0C 57624955 IC50 = 14 nM T35940 C6WO3F 57624958 IC50 = 28 nM T35940 C7JFS9 57624960 IC50 = 16 nM T35940 CYA3O4 57625005 IC50 = 63 nM T35940 CW14PM 57625015 IC50 = 99 nM T35940 CGW8C2 57652534 IC50 = 491000 nM T35940 CVK0G4 58056356 IC50 > 50000 nM T35940 CKB3A4 58102283 IC50 = 810 nM T35940 CX1G3L 58102286 IC50 = 210 nM T35940 C6BPR2 58985201 IC50 > 20000 nM T35940 C1R8NM 59139106 IC50 = 29 nM T35940 CB34LP 59139113 IC50 = 56 nM T35940 CWK9I8 59139139 IC50 = 440 nM T35940 CWN47R 59139154 IC50 = 100 nM T35940 CT0JG1 59139161 IC50 = 35 nM T35940 CP5GY6 59139172 IC50 = 190 nM T35940 CL4X3Z 59139185 IC50 = 110 nM T35940 C1PE3R 59139202 IC50 = 2900 nM T35940 CE82OV 59139228 IC50 = 44 nM T35940 C3T5OF 59139235 IC50 = 650 nM T35940 C1J2BP 59139251 IC50 = 27.7 nM T35940 CWO17Q 59139262 IC50 = 11 nM T35940 C5IYT0 59139264 IC50 = 5 nM T35940 CU3PC0 59139312 IC50 = 1190 nM T35940 C91SBH 59139388 IC50 = 940 nM T35940 C62EVK 59139472 IC50 > 50000 nM T35940 CAYO86 59229792 IC50 = 1100 nM T35940 CT3EW2 59292007 IC50 > 1000 nM T35940 CXJ63M 59603829 IC50 = 12000 nM T35940 CQEU96 59603842 IC50 = 120 nM T35940 C1MR8Q 60097495 IC50 > 10000 nM T35940 CMB3A9 66909275 IC50 = 96 nM T35940 C1UVI6 66909316 IC50 = 22 nM T35940 C37NKO 67129970 IC50 > 10000 nM T35940 CK80LJ 67130050 IC50 > 10000 nM T35940 CV63UL 67240318 IC50 > 10000 nM T35940 C7GRV2 68755406 IC50 > 10000 nM T35940 CUC21J 68796122 IC50 = 398.11 nM T35940 C5DGR9 69036886 IC50 = 10000 nM T35940 C51HSA 70791252 IC50 = 37 nM T35940 CEBO91 71452977 IC50 = 980 nM T35940 CUW41T 71460070 IC50 = 801 nM T35940 CB3SO2 71567006 IC50 > 10000 nM T35940 CDJY72 71568837 IC50 = 8600 nM T35940 CRX81Q 71575642 IC50 > 10000 nM T35940 C1AF9L 71579783 IC50 = 63 nM T35940 CGS50U 71579784 IC50 = 13 nM T35940 CIQ0N7 71579876 IC50 = 26 nM T35940 CQW94G 71579877 IC50 = 1000 nM T35940 CXC3S6 71579878 IC50 = 73 nM T35940 CG1QY4 71579965 IC50 = 76 nM T35940 C9CJR7 71579966 IC50 = 54 nM T35940 CZ31PU 71583657 IC50 > 10000 nM T35940 CXSI14 71718330 IC50 > 100000 nM T35940 C1TM3P 71720141 IC50 > 100000 nM T35940 CSVW76 72546488 IC50 = 500 nM T35940 C7HBR1 72546491 IC50 = 5 nM T35940 CXYT34 72546730 IC50 = 29 nM T35940 C1DAW5 72546731 IC50 = 21 nM T35940 C2XZW3 72708899 IC50 > 40000 nM T35940 CKN46T 72708901 IC50 > 40000 nM T35940 C2M8DV 73348939 IC50 = 157000 nM T35940 C6GZ1O 73353368 IC50 = 74 nM T35940 C7M2UX 73356583 IC50 = 25 nM T35940 C3UC9H 73891099 IC50 > 30000 nM T35940 CV8QX0 76310169 IC50 > 30000 nM T35940 CP4ZX2 76317169 IC50 = 240 nM T35940 CA5L4W 76324771 IC50 > 30000 nM T35940 C9GO0P 76328313 IC50 > 100000 nM T35940 C4DT2Z 76335375 IC50 = 85 nM T35940 C39FTZ 76335685 IC50 > 100000 nM T35940 CK61HY 85469442 IC50 = 473 nM T35940 CO2NX0 86294748 IC50 = 1.63 nM T35940 C84NEF 87200366 IC50 = 10 nM T35940 C1HW4B 89735655 IC50 = 1100 nM T35940 C6PHF1 90331409 IC50 > 10000 nM T35940 CW6S8P 90655795 IC50 > 50000 nM T35940 CNYK35 90655796 IC50 = 37000 nM T35940 CE4LR9 90655797 IC50 = 76 nM T35940 CWT2Q8 90656530 IC50 = 56.6 nM T35940 CUYE57 90656531 IC50 = 31.3 nM T35940 CENM20 90656532 IC50 = 142 nM T35940 C2DA8Y 90656533 IC50 = 101.6 nM T35940 CC3VR2 90656534 IC50 = 60.1 nM T35940 C4MN9X 90656535 IC50 = 95 nM T35940 CCJ84Q 90656536 IC50 = 112 nM T35940 C20LEX 90656537 IC50 = 123 nM T35940 CNZ8T1 90656538 IC50 = 138.5 nM T35940 C0DUR3 90656539 IC50 = 314 nM T35940 C9TUH7 90656540 IC50 = 326 nM T35940 C6BQ7R 90656541 IC50 = 411 nM T35940 CW6MU5 90656542 IC50 = 513.2 nM T35940 CW65IY 90656543 IC50 = 559 nM T35940 CUS70J 90656544 IC50 = 773 nM T35940 CU0VP1 90656545 IC50 > 1000 nM T35940 C4CI8E 90656546 IC50 > 1000 nM T35940 C3Q4ER 90656547 IC50 = 5.37 nM T35940 CK5LT8 90656548 IC50 = 11.4 nM T35940 C9JFM0 90656549 IC50 = 44.3 nM T35940 C19KMH 90656550 IC50 = 12.3 nM T35940 C8S2XK 91758407 IC50 > 10000 nM T35940 CG2Y7L 91809196 IC50 > 10000 nM T35940 C0Y8ZK 91933875 IC50 > 1000 nM T35940 C2P3LF 102136592 IC50 = 3400 nM T35940 C6AV2I 117635937 IC50 = 0.5 nM T35940 C4FIN9 117635939 IC50 = 0.019 nM T35940 C1YHR8 118633046 IC50 = 39.2 nM T35940 CLDQ03 118633052 IC50 = 57.5 nM T35940 C5BG4F 118722945 IC50 < 1000 nM T35940 CS1F8W 118722946 IC50 < 1000 nM T35940 C20GTB 118722947 IC50 < 1000 nM T35940 CJ7P1X 118723266 IC50 < 1000 nM T35940 CIH02Q 118723268 IC50 < 1000 nM T35940 C2VO8M 118723269 IC50 < 1000 nM T35940 C6VWT2 118723270 IC50 < 1000 nM T35940 CK63ST 118727694 IC50 = 27.1 nM T35940 CQCX41 118737057 IC50 > 10000 nM T35940 CE6D5X 122181354 IC50 > 1000 nM T35940 C8O7YN 122181355 IC50 > 10000 nM T35940 C8V5HL 122181356 IC50 = 4900 nM T35940 CU4ZK1 122181359 IC50 > 10000 nM T35940 C9LTM2 122181360 IC50 > 10000 nM T35940 CQ94UG 122181362 IC50 > 10000 nM T35940 CAS9U2 122181363 IC50 > 10000 nM T35940 CSON37 122181364 IC50 = 120 nM T35940 CNIA82 122181365 IC50 > 10000 nM T35940 CYDH02 122181366 IC50 = 260 nM T35940 C4X7SD 122192466 IC50 > 10000 nM T35940 CM1JW3 122604219 IC50 > 10000 nM T35940 C2UO3Y 122604256 IC50 > 10000 nM T35940 C65QNK 122604287 IC50 > 10000 nM T35940 CGT97F 122604354 IC50 > 10000 nM T35940 CW0QT8 126480560 IC50 > 10000 nM T35940 CS8C7J 126480561 IC50 > 10000 nM T35940 CCIQ37 126480562 IC50 > 10000 nM T35940 CGY2L4 126480563 IC50 > 10000 nM T35940 CJM59E 126480564 IC50 > 10000 nM T35940 CO9CY8 126480565 IC50 > 10000 nM T35940 CHQ71G 126480566 IC50 > 10000 nM T35940 C2LAM7 126591927 IC50 = 142 nM T35940 CN36JQ 127037910 IC50 = 11 nM T35940 CWL28X 127038287 IC50 = 83 nM T35940 CY95QS 127038614 IC50 = 12 nM T35940 C5S6PX 127038615 IC50 = 15 nM T35940 C04JES 127038616 IC50 = 13 nM T35940 COVZ04 127038617 IC50 = 14 nM T35940 CJ2UY6 127039306 IC50 = 22 nM T35940 CS1N3Z 127039307 IC50 = 28 nM T35940 C8C1DI 127039308 IC50 = 14 nM T35940 CB8TU5 127040913 IC50 = 18 nM T35940 CYG16V 127040980 IC50 = 15 nM T35940 CY9D7F 127040981 IC50 = 94 nM T35940 CJR5F2 127040982 IC50 = 118 nM T35940 CE0CU2 127040983 IC50 = 262 nM T35940 CUZ85G 127041304 IC50 = 345 nM T35940 CD7PL4 127041305 IC50 = 592 nM T35940 C0STZ3 127041603 IC50 = 1900 nM T35940 C58BEO 127041604 IC50 = 127 nM T35940 CUL2T4 127041605 IC50 = 15 nM T35940 CQI1H9 127041606 IC50 = 32 nM T35940 C4KZU9 127041610 IC50 = 941 nM T35940 C4S7BL 127041901 IC50 = 899 nM T35940 CZ6F5V 127042845 IC50 = 81 nM T35940 CM8J6P 127042846 IC50 = 107 nM T35940 C4NFU7 127042847 IC50 = 379 nM T35940 COZA84 127051904 IC50 = 56.7 nM T35940 C3IC2Z 127052212 IC50 = 0.015 nM T35940 C6EXU9 127052827 IC50 = 0.00715 nM T35940 CIU72D 127264586 IC50 = 161 nM T35940 C8ARK0 131801160 IC50 = 142 nM T35940 C0AV5D 131801161 IC50 = 8.5 nM T35940 CL6E4J 132601725 IC50 = 610 nM T35940 CB3C0Z 132819859 IC50 = 16 nM T35940 CK6Z5F 132819860 IC50 = 2500 nM T35940 CR3C9O 132819862 IC50 = 78 nM T35940 CAG60V 132819865 IC50 = 9.8 nM T35940 CE4Z3X 132819866 IC50 = 26 nM T35940 C8IZB3 134129887 IC50 = 4470 nM T35940 C84IXK 134130027 IC50 > 10000 nM T35940 C3TW9Y 134130036 IC50 = 8.2 nM T35940 CTDB31 134130124 IC50 = 6810 nM T35940 CZA37N 134130230 IC50 = 2480 nM T35940 C5N0CA 134130303 IC50 = 9.5 nM T35940 C4S7VK 134130361 IC50 = 1300 nM T35940 C71ATR 134130387 IC50 = 4810 nM T35940 C7U5HA 134130410 IC50 > 10000 nM T35940 C2IB7F 134130412 IC50 = 11 nM T35940 C6BCJ3 134130599 IC50 = 21 nM T35940 CH7A9R 134130612 IC50 = 763 nM T35940 CEH49U 134130924 IC50 = 8.9 nM T35940 COL93E 134131237 IC50 = 1630 nM T35940 C2AN7T 134611886 IC50 > 100000 nM T35940 CXQ03H 135413555 IC50 = 2500 nM T35940 C8GZ2B 135449326 Ki > 4000 nM T35940 C0TE5S 135651612 IC50 = 2200 nM T35940 CYDM01 135891431 IC50 > 10000 nM T35940 CM9NU1 135967827 IC50 = 32 nM T35940 C1FZ5O 135967828 IC50 = 34 nM T35940 CA0F6P 135967829 IC50 = 56 nM T35940 CM5NS2 135988101 IC50 > 2000 nM T35940 C9JH8N 135988105 IC50 > 2000 nM T35940 CZ7EX0 136183413 IC50 = 2450 nM T35940 C01QHB 137348765 IC50 = 1900 nM T35940 C7P4KI 137628642 IC50 = 10.8 nM T35940 CO19HF 137633457 IC50 > 10000 nM T35940 CI1E8V 137634241 IC50 > 10000 nM T35940 CM2VQ1 137636104 IC50 > 10000 nM T35940 CZAM24 137638642 IC50 > 10000 nM T35940 CTI5H6 137641993 IC50 > 10000 nM T35940 CCO7X8 137643676 IC50 > 10000 nM T35940 C07BXP 137644714 IC50 > 10000 nM T35940 CTDK87 137646412 IC50 > 10000 nM T35940 C7D1TY 137647232 IC50 > 10000 nM T35940 CN9A1C 137647463 IC50 > 10000 nM T35940 C5M9VT 137649141 IC50 > 10000 nM T35940 CI46SD 137652179 IC50 > 10000 nM T35940 CC32NU 137654819 IC50 > 10000 nM T35940 C6J5TG 137658266 IC50 > 10000 nM T35940 C4P2JF 137659314 IC50 > 10000 nM T35940 CS61AX 137659496 IC50 > 100000 nM T35940 CK82HJ 141401938 IC50 = 5.7 nM T35940 CKL52O 141401941 IC50 = 7.6 nM T35940 CF3RP1 141401946 IC50 = 3.9 nM T35940 CGQ16R 141401951 IC50 = 29.8 nM T35940 C14JRV 141401954 IC50 > 1000 nM T35940 C3OI7P 141401960 IC50 = 3.4 nM T35940 C89VHZ 141401969 IC50 = 21.5 nM T35940 CW1P4D 141401971 IC50 = 62.8 nM T35940 C1FIE4 145439085 IC50 = 182 nM T35940 CU62AO 145712394 IC50 = 1500 nM T35940 C6VB3O 145925651 IC50 >= 5000 nM T35940 CB06HA 145968373 IC50 > 1000 nM T35940 C73XMU 145968579 IC50 = 6 nM T35940 CQ9TX5 145968636 IC50 = 441 nM T35940 CYQF12 145970111 IC50 > 1000 nM T35940 CFU2Y5 145971060 IC50 = 7 nM T35940 CLT32B 145996530 IC50 = 100 nM T35940 C2MD1Q 155513187 IC50 > 10000 nM T35940 CUXR49 155516714 IC50 = 120 nM T35940 C4NKP6 155518298 IC50 = 1600 nM T35940 C86HPW 155518524 IC50 > 100000 nM T35940 C6EJR2 155526503 IC50 = 158.49 nM T35940 CQCL04 155545442 IC50 = 100 nM T35940 C8SU7Z 155545952 IC50 = 7.7 nM T35940 CCQ36O 155567646 IC50 = 26 nM T35940 D01WAI 135451156 IC50 = 2500 nM T35940 D06KSF 9549300 IC50 > 40000 nM T35940 D08BMM 6312649 IC50 = 2500 nM T35940 D08XVZ 24866313 IC50 > 10000 nM T35940 D0AY0F 70698427 IC50 > 10000 nM T35940 D0DQ6Z 8530 IC50 = 380 nM T35940 D0F0AX 135413546 IC50 = 2500 nM T35940 D0GD8Y 3006531 IC50 = 70 nM T35940 D0I4NN 14056555 IC50 = 2500 nM T35940 D0J3LR 11634725 Ki > 4000 nM T35940 D0M4SY 135440466 IC50 = 182 nM T35940 D0T0VC 2726555 IC50 = 7000 nM T35940 D0TF0V 3085877 IC50 = 2500 nM T35940 D0TY0P 46926364 EC50 = 4 nM T35940 D0V0QJ 389898 IC50 = 380 nM T35940 D0YE1X 9927943 IC50 > 10000 nM T67658 CO09IZ 28670291 IC50 = 20000 nM T67658 C08AQJ 42432904 IC50 = 1700 nM T67658 CM7F5P 118987010 IC50 = 195 nM T67658 C4VK7T 118987011 IC50 = 90 nM T67658 CKN7B4 135186599 IC50 = 18200 nM T67658 CRVW26 135187266 IC50 = 11000 nM T16688 D0EY0A 42636350 IC50 = 10 nM T16688 D0F1CE 53387035 IC50 = 55 nM T16688 D02NRD 9865421 IC50 = 8 nM T16688 D0F6VD 53472374 IC50 = 10 nM T16688 D0UY7A 16757107 IC50 = 38 nM T16688 D0M0NT 46926360 IC50 = 8 nM T16688 D0U5NY 10435589 IC50 = 3 nM T16688 CFN29P 1238742 IC50 = 250 nM T16688 CL21WZ 3168855 IC50 = 350 nM T16688 C3V7MF 4585845 IC50 = 1980 nM T16688 CQ0P1I 10024426 IC50 = 8 nM T16688 C8S9ZQ 10251514 IC50 = 9 nM T16688 CL3CR6 10340708 IC50 = 265 nM T16688 CO0CV2 10363180 IC50 = 8 nM T16688 CYB84U 11444140 IC50 = 73 nM T16688 C3P7AU 11502249 IC50 = 340 nM T16688 CWUS05 11538502 IC50 = 730 nM T16688 CH8AE5 11538602 IC50 = 92 nM T16688 CF90HS 11545464 IC50 = 840 nM T16688 C3IW2C 11560414 IC50 = 460 nM T16688 C57GYV 11588661 IC50 = 300 nM T16688 CP8FX4 11589415 IC50 = 190 nM T16688 C1QU0S 11603501 IC50 = 60 nM T16688 CHB92Q 11617639 IC50 = 60 nM T16688 C6IW2D 11639716 IC50 = 6.7 nM T16688 C91SGI 11646829 IC50 = 410 nM T16688 CCMV60 11660924 IC50 = 190 nM T16688 CT1L2H 11662701 IC50 = 120 nM T16688 C2HSG1 11675372 IC50 = 130 nM T16688 CR2G3N 11675641 IC50 = 460 nM T16688 C9LP6A 11690378 IC50 = 540 nM T16688 C97AKQ 11696580 IC50 = 170 nM T16688 CJK4U8 11696668 IC50 = 150 nM T16688 CE8GL2 11698356 IC50 = 35 nM T16688 CNK9X4 11703345 IC50 = 620 nM T16688 C3ZWC7 11703665 IC50 = 520 nM T16688 C1MSG2 11711001 IC50 = 350 nM T16688 CZQA97 11785312 IC50 = 81 nM T16688 CKR19P 11856514 IC50 = 8.5 nM T16688 C7B3QY 11857040 IC50 = 33 nM T16688 CER98T 13133084 IC50 = 44 nM T16688 CR26HO 15980798 IC50 = 520 nM T16688 CM48FD 15980838 IC50 = 180 nM T16688 CR56UB 15981292 IC50 = 370 nM T16688 C32OZM 15981323 IC50 = 5200 nM T16688 CSC5A8 16091082 IC50 = 320 nM T16688 C3HJ8D 16112851 IC50 = 85 nM T16688 C6AZ7J 16202164 IC50 = 15 nM T16688 CDN62P 16757011 IC50 = 160 nM T16688 CR0Z6Q 16757014 EC50 = 1500 nM T16688 CHC92G 16757105 EC50 = 490 nM T16688 C6AXO1 16757106 EC50 = 2990 nM T16688 CZ9QC1 16757108 IC50 = 48 nM T16688 CFR2A7 23624315 IC50 = 5 nM T16688 CZ0QF1 23648867 IC50 = 0.5 nM T16688 CKF7V6 23652427 IC50 = 18 nM T16688 C6Y9PU 23653376 IC50 = 4 nM T16688 CW30QM 23728888 IC50 = 3 nM T16688 CW81MR 23878093 IC50 = 130 nM T16688 CCQ56B 24768262 IC50 = 9 nM T16688 CKL21Y 24768263 IC50 = 10 nM T16688 CY8EQ0 24768264 IC50 = 11 nM T16688 C0W8RJ 24768265 IC50 = 6 nM T16688 CWVA63 24768266 IC50 = 5 nM T16688 CDC8A7 24768267 IC50 = 994 nM T16688 C4M7OE 24768269 IC50 = 35 nM T16688 CH06ZG 24768270 IC50 = 9 nM T16688 CEK35D 24768271 IC50 = 7 nM T16688 CPE7Y2 24768272 IC50 = 96 nM T16688 CQN93W 24768273 IC50 = 98 nM T16688 C94GLH 24936886 IC50 = 28000 nM T16688 CLT0O6 25016166 IC50 = 120 nM T16688 C1WLX7 25016167 IC50 = 250 nM T16688 CEZ7Y0 25016168 IC50 = 28 nM T16688 CGFM57 25016426 IC50 = 28 nM T16688 CN4XF3 25066983 IC50 = 280 nM T16688 CYFZ47 25118652 IC50 = 77 nM T16688 CKRN07 25118654 IC50 = 57 nM T16688 CG2R5L 25147516 IC50 = 64 nM T16688 CO7S3M 25174158 IC50 = 5 nM T16688 CH3L6V 25192656 IC50 = 4 nM T16688 CB0XM4 25192657 IC50 = 3 nM T16688 CA2MZ0 25192785 IC50 = 4 nM T16688 CA91JI 25196306 IC50 = 60 nM T16688 C7X6QA 25207743 IC50 = 75 nM T16688 CWPU94 25235361 IC50 = 10 nM T16688 C7URI3 25235407 IC50 = 17 nM T16688 C5MX2Q 25235717 IC50 = 47 nM T16688 CXG14U 25235767 IC50 = 23 nM T16688 CW0K5L 25235860 IC50 = 132 nM T16688 CN8DE2 36145850 IC50 = 660 nM T16688 C4K6PQ 44125987 IC50 = 100 nM T16688 C67BKX 44125988 IC50 = 520 nM T16688 CN30BK 44125989 IC50 = 110 nM T16688 CJ9L3F 44125990 IC50 = 690 nM T16688 CX0S6M 44125991 IC50 = 410 nM T16688 C52EMI 44125992 IC50 > 9100 nM T16688 C3QB0Z 44126031 IC50 = 1800 nM T16688 C6ABC7 44126032 IC50 = 310 nM T16688 C91YNG 44126033 IC50 = 30 nM T16688 CL27CS 44126034 IC50 = 170 nM T16688 CZ19XD 44126083 IC50 = 60 nM T16688 C9C2NE 44126086 IC50 = 1100 nM T16688 C75QFI 44444912 IC50 = 9 nM T16688 CDX1E5 44464393 IC50 = 73 nM T16688 C4TM5S 44565367 IC50 = 69 nM T16688 C9OLR5 46208314 IC50 = 79 nM T16688 CN3BE0 46212588 IC50 = 41 nM T16688 C9IM6Q 46843707 IC50 = 600 nM T16688 CUL91T 46843708 IC50 = 16 nM T16688 CT4AW3 46843774 IC50 = 29 nM T16688 CVR63G 46843777 IC50 = 162 nM T16688 CR8KH0 46843840 IC50 = 1190 nM T16688 CW2XB8 46843841 IC50 = 70 nM T16688 CHOT17 46843842 IC50 = 66 nM T16688 CK4Y2X 46843843 IC50 = 181 nM T16688 CP6DF7 46843845 IC50 = 970 nM T16688 CCP3T1 46843909 IC50 = 4770 nM T16688 CZ4DU8 46843911 IC50 = 838 nM T16688 CF92ZP 46843912 IC50 = 44 nM T16688 CW89AO 46843913 IC50 = 33 nM T16688 CD17CQ 46847261 IC50 = 38 nM T16688 CZC06K 46847559 IC50 = 1390 nM T16688 C57LYQ 46849596 IC50 = 134 nM T16688 CAX57D 46850597 IC50 = 60 nM T16688 CO34ZH 46850971 IC50 = 82 nM T16688 C2Y9LH 46850972 IC50 = 142 nM T16688 CNMB07 46851121 IC50 = 426 nM T16688 CCH12P 46851123 IC50 = 12 nM T16688 CI59YE 46851124 IC50 = 498 nM T16688 CEJW98 46851125 IC50 = 47 nM T16688 CQKB14 46851126 IC50 = 85 nM T16688 CJ8VO6 46851466 IC50 = 45 nM T16688 CX1E2G 46851467 IC50 = 55 nM T16688 CA0E6S 46851790 IC50 = 40 nM T16688 C2V8IH 46851792 IC50 = 218 nM T16688 CU36HJ 46851954 IC50 = 350 nM T16688 C78SZA 46851956 IC50 = 2840 nM T16688 CFK65J 46852111 IC50 = 1190 nM T16688 C67PWE 46852113 IC50 = 12 nM T16688 CYRX62 46852114 IC50 = 233 nM T16688 C3KZU8 46852423 IC50 = 92 nM T16688 CVA1C2 46852425 IC50 = 81 nM T16688 C86BDJ 46852578 IC50 = 122 nM T16688 CRH68F 46852579 IC50 = 279 nM T16688 CYFZ49 46852580 IC50 = 88 nM T16688 CQ6IP3 46852727 IC50 = 11 nM T16688 CJQ7V4 46852730 IC50 = 408 nM T16688 CIB91O 46852883 IC50 = 9 nM T16688 CX58NY 46865791 IC50 = 22 nM T16688 C1F4RW 46884873 IC50 = 650 nM T16688 CK0VG9 46884874 IC50 = 2000 nM T16688 CWP5A9 46884916 IC50 = 220 nM T16688 CWFS79 46884917 IC50 = 790 nM T16688 CO4GB6 46884918 IC50 = 94 nM T16688 CDI0G1 46884919 IC50 = 140 nM T16688 CZK9Y5 46884949 IC50 = 44 nM T16688 CJ6CE2 46884950 IC50 = 28 nM T16688 CVI3U4 46884951 IC50 = 1900 nM T16688 CSN6J8 46884952 IC50 = 5500 nM T16688 C07YJN 46885000 IC50 = 98 nM T16688 CH2YB8 46885001 IC50 > 10000 nM T16688 CLY1F5 46885002 IC50 > 10000 nM T16688 CBW54P 46885003 IC50 > 10000 nM T16688 CCV8Q2 46885136 IC50 > 10000 nM T16688 CRG47E 46885137 IC50 = 5300 nM T16688 C9ZJ4B 46885138 IC50 = 2800 nM T16688 CKFM62 46885139 IC50 = 3600 nM T16688 C0B3EF 46885188 IC50 = 79 nM T16688 C9GDC3 46885189 IC50 = 1300 nM T16688 CD3T8U 46885190 IC50 = 49 nM T16688 C95MOI 46885191 IC50 = 25 nM T16688 C38HZR 46885246 IC50 = 700 nM T16688 C7OJ0Z 46897950 IC50 = 12 nM T16688 CM8EH2 46926717 IC50 = 100 nM T16688 CRF5N9 46926794 IC50 = 275 nM T16688 CCY12P 46946735 IC50 = 37 nM T16688 C8VOS1 46946932 IC50 = 56 nM T16688 CRH93W 49800157 IC50 = 19 nM T16688 C2J9TU 49800160 IC50 < 30 nM T16688 C9L3XR 49838879 IC50 > 20000 nM T16688 CB74WR 49846142 IC50 = 12.59 nM T16688 C7W9XS 49846145 IC50 = 19.95 nM T16688 CIK51U 49846226 IC50 = 3.981 nM T16688 CTSA42 49847173 IC50 = 6.31 nM T16688 C5W7AQ 52916959 IC50 = 280 nM T16688 C3WXY8 52916960 IC50 = 311 nM T16688 CU0DG3 52917199 IC50 = 344 nM T16688 C9HJ6X 52917342 IC50 = 482 nM T16688 CZ63IA 52917345 IC50 = 125 nM T16688 CL0GA3 52917417 IC50 = 70 nM T16688 C2W3TR 52917419 IC50 = 145 nM T16688 CAWY86 52917420 IC50 = 55 nM T16688 CQI39M 52917491 IC50 = 51 nM T16688 C7Y4UD 52917492 IC50 = 60 nM T16688 CJL3M5 52917495 IC50 = 194 nM T16688 CJ1PU8 52917631 IC50 = 25 nM T16688 CF1ZP5 52917632 IC50 = 33 nM T16688 COF60B 52917633 IC50 = 39 nM T16688 C3X6BV 52917634 IC50 = 24 nM T16688 C3SL4W 52917635 IC50 = 42 nM T16688 CW6EA0 52917768 IC50 = 52 nM T16688 CE9L1O 52917770 IC50 = 103 nM T16688 C7VGW8 52917838 IC50 = 774 nM T16688 C1QY6K 52936629 IC50 = 15100 nM T16688 CYZ0G1 52936630 IC50 = 24700 nM T16688 COH9G0 52936726 EC50 = 1803 nM T16688 CUFQ14 52936727 EC50 = 228 nM T16688 C9Q3RD 52936729 EC50 = 25000 nM T16688 C0QFD5 52936730 IC50 = 202 nM T16688 C1ND6F 52936731 EC50 = 138 nM T16688 CI5P2Z 52936838 EC50 = 216 nM T16688 C92MVO 52936839 IC50 = 41 nM T16688 CH3OR6 52936840 EC50 = 410 nM T16688 C4CU6Y 52936841 EC50 = 378 nM T16688 CF0ZV9 52936842 EC50 = 219 nM T16688 CK94GN 52936952 IC50 = 136 nM T16688 C6AJP0 52936953 EC50 = 190 nM T16688 CZ9N4K 52936954 EC50 = 362 nM T16688 C05OXZ 52936955 EC50 = 371 nM T16688 CMV72X 52936956 EC50 = 1764 nM T16688 C4PQ8A 52937057 EC50 = 2363 nM T16688 CT05UL 52940751 IC50 = 110 nM T16688 COQ10T 52941984 IC50 = 160 nM T16688 CNK5E8 52941985 IC50 > 3000 nM T16688 CI0YM9 52942491 IC50 = 630 nM T16688 C7N5PG 52942592 IC50 > 1000 nM T16688 C3ALM2 52942635 IC50 = 250 nM T16688 C7K4OU 52942652 IC50 = 520 nM T16688 CZU29W 52942808 IC50 = 56 nM T16688 CB0Q3W 52943161 IC50 > 3000 nM T16688 CJQP92 52943202 IC50 = 220 nM T16688 CN6B7T 52943363 IC50 = 380 nM T16688 CCP4D9 52943384 IC50 > 1000 nM T16688 C7KYL1 52943385 IC50 = 240 nM T16688 CGS1W6 52943386 IC50 = 65 nM T16688 C4XE3I 52943771 IC50 = 830 nM T16688 C8U6MZ 52943823 IC50 = 60 nM T16688 C3G6SY 52943844 IC50 = 570 nM T16688 C3KQG6 52943853 IC50 > 3000 nM T16688 CCS5X0 52944039 IC50 > 3000 nM T16688 CE9L0P 52944382 IC50 > 3000 nM T16688 C6KQ1W 52944897 IC50 > 3000 nM T16688 CP9R2G 52945115 IC50 = 470 nM T16688 CTG39K 52945136 IC50 = 290 nM T16688 C9J7GN 52945149 IC50 = 120 nM T16688 CO5T6P 52945817 IC50 = 620 nM T16688 CIR7X5 52946164 IC50 = 1360 nM T16688 C57IQK 52946165 IC50 = 120 nM T16688 CS9Z8D 52946166 IC50 = 180 nM T16688 C35GAK 52946243 IC50 > 3000 nM T16688 CDJG27 52946271 IC50 = 270 nM T16688 CE6D8X 52946281 IC50 = 290 nM T16688 CJ3X5Y 52946365 IC50 = 68 nM T16688 CMZ6P0 52946512 IC50 = 51 nM T16688 C2HNM3 52947394 IC50 = 140 nM T16688 CB38OM 52947444 IC50 = 69 nM T16688 C24EOF 52947585 IC50 = 200 nM T16688 CBD4T3 52947757 IC50 = 240 nM T16688 CUHW67 52948237 IC50 = 2500 nM T16688 CMI8J0 52948238 IC50 = 110 nM T16688 C7HN3L 52948573 IC50 = 100 nM T16688 C6HZ5R 52948779 IC50 = 110 nM T16688 CMBC05 52949863 IC50 = 6100 nM T16688 CKA56O 52949871 IC50 = 270 nM T16688 CQ36FR 52950072 IC50 = 52 nM T16688 CX17CT 53326694 IC50 = 14 nM T16688 C7D5TK 53389580 IC50 = 19.95 nM T16688 C6GS7N 53472377 IC50 = 10 nM T16688 CCUA63 53472426 IC50 = 39.81 nM T16688 CV8N6Y 53472427 IC50 = 63.1 nM T16688 CXO59S 53472469 IC50 = 79.43 nM T16688 C4R6IL 53472470 IC50 = 19.95 nM T16688 CD5JT0 53472471 IC50 = 50.12 nM T16688 C3UY7X 53472473 IC50 = 50.12 nM T16688 CZ05VY 53484046 IC50 = 17 nM T16688 C8DNF3 53484047 IC50 = 14 nM T16688 C7PC9D 53484048 IC50 = 14 nM T16688 CNC9V1 53484049 IC50 = 18 nM T16688 C5CE4L 53484071 IC50 = 25 nM T16688 CLPB05 54580056 IC50 = 44 nM T16688 C50QHE 54580057 IC50 = 7 nM T16688 C0AND9 54582083 IC50 = 237 nM T16688 CSKW81 54754161 IC50 = 10 nM T16688 CE6Z4W 56602801 IC50 = 137 nM T16688 CUJ89T 56602861 IC50 = 301 nM T16688 CR4I1O 56602863 IC50 = 68 nM T16688 CFVR29 56602864 IC50 = 377 nM T16688 CNBS87 56602865 IC50 = 330 nM T16688 C91PGO 56603115 IC50 = 19 nM T16688 C5ES6P 56603116 IC50 = 6 nM T16688 CVI51O 56603118 IC50 = 10 nM T16688 C2IM6T 56603174 IC50 = 19 nM T16688 CH05TN 56603175 IC50 = 18 nM T16688 CFXG65 56603176 IC50 = 6 nM T16688 CDL94H 56603301 IC50 = 24 nM T16688 C9D1MV 56603353 IC50 = 23 nM T16688 C60YTB 56603356 IC50 = 3 nM T16688 CZM92Q 56603411 IC50 = 52 nM T16688 C52EWD 56603412 IC50 = 137 nM T16688 CJVR02 56603413 IC50 = 10 nM T16688 CUM63A 56603464 IC50 = 66 nM T16688 CN5QZ2 56645797 IC50 = 286 nM T16688 C4NR3W 56645798 IC50 = 253 nM T16688 CZ1XD9 56645800 IC50 = 57 nM T16688 CW1X7R 56645990 IC50 = 120 nM T16688 CWE6L8 56658045 IC50 = 30 nM T16688 C6HI2C 56658046 IC50 = 72 nM T16688 CX9C4O 56664974 IC50 = 32 nM T16688 CY56CN 56668305 IC50 = 225 nM T16688 CZM86Q 56668406 IC50 = 28 nM T16688 C7R6FV 56668407 IC50 = 99 nM T16688 CTS5V9 56671786 IC50 = 175 nM T16688 CE76DX 56671915 IC50 = 57 nM T16688 CVO6G3 56675292 IC50 = 88 nM T16688 CJ0EC7 56678494 IC50 = 98 nM T16688 C6KFW9 56678757 IC50 = 64 nM T16688 CKI9P1 56681839 IC50 = 245 nM T16688 CXDC48 56681956 IC50 = 51 nM T16688 CB35ES 56682061 IC50 = 18 nM T16688 CSQ8J7 56839306 IC50 = 116 nM T16688 CNGF94 56839506 IC50 = 460 nM T16688 CO5B2H 56839731 IC50 = 54 nM T16688 CBHT83 56840376 IC50 = 29 nM T16688 CV8W4T 56933229 IC50 = 8 nM T16688 C75IPK 56950373 IC50 = 49 nM T16688 C69NBW 56950374 IC50 = 102 nM T16688 CAV46L 56950511 IC50 = 97 nM T16688 CT01DK 56950512 IC50 = 167 nM T16688 CA0UD3 56959088 IC50 = 3.5 nM T16688 CTBQ39 56959224 IC50 = 2.3 nM T16688 C0IO6U 56959226 IC50 = 1.7 nM T16688 CPFX65 56960522 IC50 = 1.1 nM T16688 CBAZ68 57326908 IC50 = 1860 nM T16688 C9LD6E 57326909 IC50 > 10000 nM T16688 C76EDM 57326910 IC50 > 10000 nM T16688 CZ5HX4 57326911 IC50 = 250 nM T16688 CK2RY3 57326912 IC50 = 110 nM T16688 C1IQK6 57326913 IC50 > 10000 nM T16688 CZ7F9E 57326914 IC50 > 10000 nM T16688 CMR6I7 57328828 IC50 = 110 nM T16688 CW60MQ 57390208 IC50 = 230 nM T16688 CZ24WT 57391495 IC50 = 330 nM T16688 C4G6HE 57391496 EC50 = 910 nM T16688 CY45KB 57393260 EC50 = 8090 nM T16688 C6PX4J 57393261 EC50 = 8900 nM T16688 C35VYF 57393687 IC50 = 520 nM T16688 CMG4H2 57393709 IC50 = 11 nM T16688 C1VFZ7 57393718 IC50 = 4 nM T16688 CG2XP3 57393719 IC50 = 29 nM T16688 CGY74E 57394982 IC50 = 43000 nM T16688 CKB53U 57395435 IC50 = 144 nM T16688 C8X7NR 57395436 IC50 = 39 nM T16688 CROM50 57395437 IC50 = 117 nM T16688 C9FMZ1 57397247 IC50 = 2420 nM T16688 CSJQ04 57397275 IC50 = 13 nM T16688 CE7G9Q 57397280 IC50 = 110 nM T16688 C1W9FP 57397281 IC50 = 53 nM T16688 CE0I6B 57397282 IC50 = 373 nM T16688 CDVW75 57398504 EC50 = 3700 nM T16688 C8WN9M 57398505 IC50 = 699 nM T16688 CVK9Y3 57398514 IC50 = 9900 nM T16688 C25YSQ 57398966 IC50 = 20 nM T16688 CS7J8Y 57398967 IC50 = 1120 nM T16688 C9YKL3 57400676 IC50 = 38 nM T16688 CC7QY8 57401961 EC50 = 3420 nM T16688 CZD1R2 57401962 EC50 = 7460 nM T16688 CVC2F5 57401980 IC50 = 7400 nM T16688 CT34CJ 57402458 IC50 = 28 nM T16688 CX1YQ3 57402459 IC50 = 115 nM T16688 CX4MW2 57403714 IC50 = 407 nM T16688 CRX48M 57403734 IC50 = 13900 nM T16688 CA1X0O 57404460 IC50 = 30 nM T16688 C7GYW4 57404461 IC50 = 35 nM T16688 CE2W7D 57404462 IC50 = 30 nM T16688 C5P3HT 57545640 IC50 = 1327 nM T16688 C10CAG 57991984 IC50 = 6309.57 nM T16688 C1ET5C 57992001 IC50 = 41000 nM T16688 CH3YR2 57992005 IC50 > 10000 nM T16688 CEI9W6 57992028 IC50 = 1900 nM T16688 C7CAE9 57992030 IC50 = 60 nM T16688 C52VNA 57992036 IC50 = 110 nM T16688 C2Z8GJ 57992039 IC50 = 590 nM T16688 C0U9MB 57992045 IC50 = 6309.57 nM T16688 CCH4G6 57992058 IC50 = 200 nM T16688 C5DWU9 57992078 IC50 = 80 nM T16688 CUKI92 57992081 IC50 = 30 nM T16688 CJ7HL3 57992094 IC50 = 125.89 nM T16688 CS19RN 57992122 IC50 = 60000 nM T16688 CXB17A 57992140 IC50 = 1200 nM T16688 C8VOZ4 57992168 IC50 = 630.96 nM T16688 C47UAO 57992175 IC50 = 30 nM T16688 C5J3AP 57992180 IC50 = 100 nM T16688 C6OQF9 57992190 IC50 = 1100 nM T16688 C37TMQ 57992198 IC50 = 1900 nM T16688 C0B6DH 57992215 IC50 = 120 nM T16688 C0QMK7 58064355 IC50 = 52 nM T16688 CAS3R5 58064386 IC50 = 3100 nM T16688 CQ23XC 58064402 IC50 > 10000 nM T16688 CS5HB3 58064415 IC50 = 2393 nM T16688 CVQ01T 58064420 IC50 = 20 nM T16688 CZ4IS5 58064430 IC50 = 11 nM T16688 C8S5AN 58064438 IC50 > 10000 nM T16688 C6Y9VQ 58064440 IC50 = 33 nM T16688 C48WXN 58064443 IC50 > 10000 nM T16688 CC05UV 58064451 IC50 = 2735 nM T16688 C65VET 58064459 IC50 = 41 nM T16688 C2SF5Y 58064473 IC50 > 10000 nM T16688 C6T2HE 58064474 IC50 = 1900 nM T16688 CFP23X 58064480 IC50 = 91 nM T16688 C6MO8E 58064492 IC50 > 10000 nM T16688 C28RCD 58064510 IC50 = 450 nM T16688 CF8WS2 58064515 IC50 = 950 nM T16688 CL9V6F 58064516 IC50 > 10000 nM T16688 CWA89N 58064526 IC50 = 69 nM T16688 C5EQI0 58064529 IC50 = 2900 nM T16688 CU6KM8 58064531 IC50 = 110 nM T16688 CJ5U7P 58064536 IC50 = 5548 nM T16688 CX1B7D 58064544 IC50 = 360 nM T16688 CHS70X 58064553 IC50 = 560 nM T16688 C3PC2S 58064559 IC50 > 10000 nM T16688 C7D9WZ 58064580 IC50 > 10000 nM T16688 CDVL20 58064582 IC50 = 20 nM T16688 C3W8MT 58064604 IC50 = 6100 nM T16688 C4DLM1 58064608 IC50 = 160 nM T16688 CC1K6S 58064620 IC50 = 28 nM T16688 CCF8N3 58064672 IC50 = 300 nM T16688 CBDM27 58064687 IC50 > 10000 nM T16688 CP0C1K 58230907 IC50 = 6 nM T16688 C3BVX1 58230968 IC50 = 5 nM T16688 CCZ0V6 58428904 IC50 = 79 nM T16688 C1CVR4 58464413 IC50 = 7.7 nM T16688 C34UQR 58464414 IC50 = 31.62 nM T16688 CG68OA 58464429 IC50 = 25.12 nM T16688 C51EZB 58464432 IC50 = 39.81 nM T16688 C3M9XN 58464439 IC50 = 79.43 nM T16688 C5GF9H 58464441 IC50 = 15.85 nM T16688 CR4OJ7 58464474 IC50 = 15.85 nM T16688 CBT53K 58464475 IC50 = 25.12 nM T16688 C7EK6J 58464480 IC50 = 19.95 nM T16688 CA9E1G 58464487 IC50 = 50.12 nM T16688 CYBN91 58464510 IC50 = 15.85 nM T16688 CI9H3Y 58464524 IC50 = 39.81 nM T16688 CQE02I 58464533 IC50 = 50.12 nM T16688 CJ4ZX7 58464537 IC50 = 251.19 nM T16688 CV39OR 58577911 IC50 = 640 nM T16688 CRK7G6 58577912 IC50 = 410 nM T16688 CXT24F 58909524 IC50 = 20 nM T16688 CYX32E 58909548 IC50 = 2500 nM T16688 C15SPI 58909560 IC50 = 15 nM T16688 C47XIB 58909583 IC50 = 50 nM T16688 CMX8H1 58909584 IC50 > 10000 nM T16688 CS79EG 58909599 IC50 = 6 nM T16688 CUJL48 58909623 IC50 = 160 nM T16688 CBVA73 58909630 IC50 = 610 nM T16688 C7UKR3 58909641 IC50 = 3300 nM T16688 CXJR91 58909657 IC50 = 810 nM T16688 CB3JQ6 58909669 IC50 > 10000 nM T16688 C1GWH2 58909670 IC50 = 7500 nM T16688 C8GD5H 58909676 IC50 = 2900 nM T16688 CL6D1M 58909690 IC50 = 490 nM T16688 CAJ06H 58909701 IC50 = 390 nM T16688 C7A4DB 58909703 IC50 = 210 nM T16688 CYIQ86 58909704 IC50 = 5900 nM T16688 CSKO67 58909722 IC50 = 580 nM T16688 CGKC98 58909735 IC50 = 50 nM T16688 CGDM34 58909745 IC50 = 220 nM T16688 CQ92BD 58909750 IC50 = 5 nM T16688 CEW7J8 58909754 IC50 = 390 nM T16688 CGTE96 58909771 IC50 = 150 nM T16688 CYL3O4 58909777 IC50 = 90 nM T16688 CT5UA8 58909801 IC50 = 130 nM T16688 C87QFK 58909803 IC50 = 410 nM T16688 C2OR1B 58909807 IC50 = 6 nM T16688 CZI9L0 58909815 IC50 = 570 nM T16688 CV0IB3 58909821 IC50 = 50 nM T16688 CZ3T8O 58909823 IC50 = 390 nM T16688 CNP31S 58909825 IC50 = 120 nM T16688 C26MGP 58909844 IC50 = 60 nM T16688 CXSQ61 58909847 IC50 > 10000 nM T16688 CM2DK7 58909856 IC50 = 10 nM T16688 C2PO1S 58909858 IC50 = 470 nM T16688 C4MD6H 58909862 IC50 = 90 nM T16688 CO1KX8 58909929 IC50 > 10000 nM T16688 C0SD1I 59302499 IC50 = 76 nM T16688 CST3M6 59302503 IC50 = 34 nM T16688 CJA98G 59302536 IC50 = 8 nM T16688 C7D8PS 59440849 IC50 = 25 nM T16688 C7TQ1N 59440858 IC50 = 40 nM T16688 CFX1N3 59440860 IC50 = 45 nM T16688 CJMS68 59440876 IC50 = 210 nM T16688 CH8U9K 59440882 IC50 = 185 nM T16688 CP5W1Q 59440891 IC50 = 312 nM T16688 C03EFU 59440893 IC50 = 60 nM T16688 CG4I8D 59440898 IC50 = 609 nM T16688 CDCU41 59440900 IC50 = 253 nM T16688 C0J4HN 59464134 IC50 = 120 nM T16688 C29WMR 59464136 IC50 = 7 nM T16688 CHR64M 59464293 IC50 > 30000 nM T16688 CS3G6Y 59464296 IC50 = 5.7 nM T16688 C14IKC 59464318 IC50 = 3300 nM T16688 CZC8Y2 59464331 IC50 = 4.4 nM T16688 CXC7L2 59627660 IC50 = 25.12 nM T16688 CWF35C 59627683 IC50 = 7.943 nM T16688 C45XVN 60142198 IC50 = 4.5 nM T16688 CJ5M9S 60142200 IC50 = 4.5 nM T16688 C79ZOY 60142335 IC50 = 2.5 nM T16688 C32XVA 60150582 IC50 = 39 nM T16688 CG1SO5 66677706 IC50 = 1700 nM T16688 CMYH02 66677711 IC50 = 180 nM T16688 C5FQI0 66678194 IC50 = 630 nM T16688 C3U0YB 66678231 IC50 = 2030 nM T16688 C86DMW 66678414 IC50 = 3100 nM T16688 C9H6FG 66739879 IC50 = 48 nM T16688 CNEW29 66740330 IC50 = 5280 nM T16688 CD4ZN9 66740435 IC50 = 144 nM T16688 C3QVI2 66965549 IC50 = 56 nM T16688 C2VR8T 66965566 IC50 = 500 nM T16688 CYD84R 66965700 IC50 = 28 nM T16688 CQ0BA9 66965879 IC50 = 1400 nM T16688 CMAG74 66965885 IC50 = 28 nM T16688 CD8XN4 66966108 IC50 = 32 nM T16688 CF1C8W 67027009 IC50 = 32 nM T16688 CIE7S3 67035798 IC50 = 40 nM T16688 CFL4C7 67035960 IC50 = 152 nM T16688 CL36VN 67293479 IC50 = 66 nM T16688 C7LKN0 67293543 IC50 = 1508 nM T16688 C9M7JW 67293558 IC50 = 93 nM T16688 CO6L7T 67293617 IC50 = 228 nM T16688 CU13AW 67293628 IC50 = 6870 nM T16688 C7MHS8 67293664 IC50 = 79 nM T16688 CCF16H 67293673 IC50 = 4749 nM T16688 CUD4I7 67293707 IC50 = 1708 nM T16688 C0O2YR 67293853 IC50 = 938 nM T16688 C89JDW 67336578 IC50 = 125.89 nM T16688 CWN3Q2 67336857 IC50 = 316.23 nM T16688 C4KZ6M 67387006 IC50 = 513 nM T16688 C50IMJ 67387021 IC50 = 41 nM T16688 CI4OM6 67389970 IC50 = 3870 nM T16688 CCQL14 67390528 IC50 = 180 nM T16688 CF4KW9 67390709 IC50 = 46 nM T16688 C7RI4N 67391714 IC50 = 67 nM T16688 CUR27D 67408586 IC50 = 474 nM T16688 CZ60KP 67436594 IC50 = 50.12 nM T16688 CU2CP1 67437893 IC50 = 39.81 nM T16688 C10UPR 67437917 IC50 = 31.62 nM T16688 C4ZQT7 67439764 IC50 = 50.12 nM T16688 CWD2N8 67995764 IC50 = 860 nM T16688 CX0ER3 68007164 IC50 = 240 nM T16688 C2NOD0 68038529 IC50 = 41 nM T16688 C4K0LV 68038557 IC50 = 149 nM T16688 C2ULQ3 68046818 IC50 = 17 nM T16688 CBOF40 68046989 IC50 = 10 nM T16688 CR05NW 68083430 IC50 = 7257 nM T16688 CG54WP 68235801 IC50 = 631 nM T16688 CHM8N2 68235802 IC50 = 1381 nM T16688 CU2LC9 68235882 IC50 = 788 nM T16688 C5D0UM 68236004 IC50 = 311 nM T16688 CTJ4V2 68236190 IC50 = 731 nM T16688 C3US5Z 68236199 IC50 = 5837 nM T16688 CY9V7N 68581205 IC50 = 94 nM T16688 CCQ1Z4 68581919 IC50 = 44 nM T16688 C2NGS5 68582100 IC50 = 13 nM T16688 CJZ7K3 68582726 IC50 = 32 nM T16688 CLE65O 68681268 IC50 = 80 nM T16688 C0FZ8A 68682128 IC50 = 210 nM T16688 CSXO57 68682453 IC50 = 23 nM T16688 CHV46B 68682544 IC50 = 1300 nM T16688 C8ING5 68682560 IC50 = 540 nM T16688 CE4D6H 68682592 IC50 = 16 nM T16688 CRE6O1 68682846 IC50 = 3 nM T16688 CH86IV 68682918 IC50 = 13 nM T16688 C4MK8Y 68683665 IC50 = 32 nM T16688 CI34YM 68683791 IC50 = 70 nM T16688 C6Y7XF 68685264 IC50 = 620 nM T16688 CTU49O 68685968 IC50 = 6.6 nM T16688 C8QS0B 68686037 IC50 = 310 nM T16688 CJV84X 68686074 IC50 = 35 nM T16688 C5ZSV0 70355830 IC50 = 10.2 nM T16688 C6RC4J 70681764 IC50 = 3700 nM T16688 C42FXK 70681777 IC50 = 2100 nM T16688 CW2LD6 70686525 IC50 = 1300 nM T16688 C34GTB 70688145 IC50 = 1300 nM T16688 C03QWH 70689493 IC50 > 10000 nM T16688 CD1E8K 70690180 IC50 > 30000 nM T16688 C0YD8S 70691611 IC50 = 65 nM T16688 CVZB58 70691612 IC50 = 30 nM T16688 CFP4L8 70691613 IC50 > 10000 nM T16688 CR3G1D 70693693 IC50 > 10000 nM T16688 CEH95V 70693694 IC50 = 2360 nM T16688 CNV13L 70694391 IC50 = 11000 nM T16688 CZ5D3I 70694392 IC50 = 8000 nM T16688 CJ87BY 71061220 IC50 = 50 nM T16688 CA3S7F 71061400 IC50 = 6 nM T16688 C14UHB 71061524 IC50 = 126 nM T16688 C7J3GS 71061548 IC50 = 63 nM T16688 CPUX27 71061587 IC50 = 200 nM T16688 C0WKU5 71061589 IC50 = 16 nM T16688 C43HIW 71061665 IC50 = 2 nM T16688 CDS8I7 71061693 IC50 = 32 nM T16688 CCMX86 71061697 IC50 = 63 nM T16688 CXM2H9 71061713 IC50 = 3 nM T16688 CC29LF 71061726 IC50 = 63 nM T16688 C7K9TL 71061822 IC50 = 5100 nM T16688 CRX68H 71062784 IC50 = 16 nM T16688 C4MD6K 71062800 IC50 = 2820 nM T16688 CNX19G 71062856 IC50 = 32 nM T16688 C39RAY 71063102 IC50 = 3 nM T16688 C6HRB4 71077940 IC50 = 6.5 nM T16688 C6NKY5 71078482 IC50 = 5.8 nM T16688 C50WGF 71078515 IC50 = 2.5 nM T16688 CK3UR0 71080439 IC50 = 2.5 nM T16688 CM2UF1 71080444 IC50 = 20 nM T16688 CVF7J3 71080446 IC50 = 10 nM T16688 C9AUY0 71080447 IC50 = 16 nM T16688 CK83IL 71080489 IC50 = 126 nM T16688 CFK50V 71110267 IC50 = 3.1 nM T16688 CS4T0U 71110270 IC50 = 2.2 nM T16688 C3ORQ5 71110347 IC50 = 2 nM T16688 CIX83R 71110421 IC50 = 61.3 nM T16688 CW7N8M 71110422 IC50 = 442.5 nM T16688 C3G7QB 71110423 IC50 = 23.6 nM T16688 CD80YI 71110425 IC50 = 50.5 nM T16688 CAH09S 71110518 IC50 = 15.2 nM T16688 CRW60H 71110609 IC50 = 2 nM T16688 CN45QO 71217314 IC50 = 540 nM T16688 CX9K0J 71449800 IC50 = 1580 nM T16688 C5JF6C 71453442 IC50 > 10000 nM T16688 C87NDY 71453680 IC50 = 40 nM T16688 C51KBV 71455455 IC50 > 10000 nM T16688 C3PU7T 71457189 IC50 > 10000 nM T16688 CQA32X 71459046 IC50 > 33000 nM T16688 CAC7W5 71460852 IC50 = 120 nM T16688 CR2V9E 71462556 IC50 > 10000 nM T16688 C1HWI0 71462595 IC50 > 10000 nM T16688 COI42Y 71478198 IC50 = 26.1 nM T16688 CDSK92 71534758 IC50 = 30.3 nM T16688 CU7C4H 71534759 IC50 = 3.5 nM T16688 CD7B2I 71534760 IC50 = 15.9 nM T16688 CYWR98 71534761 IC50 = 18.4 nM T16688 CFJB93 71535057 IC50 = 32.1 nM T16688 CWL0K3 71538697 IC50 = 23.4 nM T16688 CQX6G0 71538698 IC50 = 39.9 nM T16688 CHX21Q 71538699 IC50 = 8.5 nM T16688 CNE85M 71538700 IC50 = 3.7 nM T16688 COF38Y 71538701 IC50 = 8.8 nM T16688 C9D6XL 71538702 IC50 = 59.2 nM T16688 CN8U3X 71552011 IC50 = 190 nM T16688 C7QV1A 71552091 IC50 = 120 nM T16688 C58ZCX 71552092 IC50 = 392 nM T16688 CY08FK 71571356 IC50 > 10000 nM T16688 C4R3WA 71571718 IC50 = 2 nM T16688 C6SU2O 71572050 IC50 = 11.6 nM T16688 C14BCP 71572051 IC50 = 7 nM T16688 CB1YS4 71572385 IC50 = 30.8 nM T16688 CR0KX9 71572386 IC50 = 3.6 nM T16688 CN52ZY 71572387 IC50 = 3.2 nM T16688 C49QLP 71602372 IC50 > 10000 nM T16688 CR13XU 71602433 IC50 > 10000 nM T16688 C38SOR 71602434 IC50 > 10000 nM T16688 C3ZR8K 71603028 IC50 > 10000 nM T16688 CP97OC 71603093 IC50 > 10000 nM T16688 CAHY94 71603095 IC50 > 10000 nM T16688 C3IHF5 71603097 IC50 > 10000 nM T16688 CQ1K6W 71603210 IC50 > 10000 nM T16688 C9D1QC 71603211 IC50 > 10000 nM T16688 C8JKL2 71603212 IC50 > 10000 nM T16688 CEB4W2 71717630 IC50 = 119 nM T16688 C73WPT 71730102 IC50 = 9.6 nM T16688 C7Z1IR 71730238 IC50 = 0.7 nM T16688 CF78GV 71730361 IC50 = 1.3 nM T16688 CFHK37 71730881 IC50 = 98 nM T16688 CNH38L 71731010 IC50 = 127 nM T16688 CPB1F0 71731512 IC50 = 6.4 nM T16688 CQ82DI 71731513 IC50 = 38 nM T16688 CJTR16 71766152 IC50 > 50000 nM T16688 C0DSR2 71769147 IC50 = 274 nM T16688 CQ97XH 71769148 IC50 = 85 nM T16688 CE4T3O 71769149 IC50 = 470 nM T16688 CN40OE 71769150 IC50 = 113 nM T16688 CD72ET 71769151 IC50 = 6750 nM T16688 CQW5G0 71769152 IC50 = 88 nM T16688 CS65TV 71769281 IC50 = 79 nM T16688 CXU7E1 71769282 IC50 = 174 nM T16688 C5PTF4 71769396 IC50 = 70 nM T16688 CHB7Z4 71770420 IC50 = 2960 nM T16688 CMH20C 71770421 IC50 > 3000 nM T16688 C25JOU 71770539 IC50 > 3000 nM T16688 C3S5XH 71770540 IC50 > 3000 nM T16688 CD5H2L 71770541 IC50 > 3000 nM T16688 C4PC0Z 71770542 IC50 > 3000 nM T16688 C8Z5TF 71770543 IC50 = 1200 nM T16688 C8OKJ0 71770544 IC50 = 23 nM T16688 C24FIU 71770664 IC50 = 625 nM T16688 CSD58Z 71770666 IC50 = 681 nM T16688 C0H5CU 71770668 IC50 = 92100 nM T16688 C5FAP9 71770669 IC50 = 2950 nM T16688 C9F8UJ 71770784 IC50 = 31 nM T16688 CJAX51 71770785 IC50 = 26 nM T16688 CN1PI0 71770909 IC50 = 68 nM T16688 C6B1TS 71770910 IC50 = 55 nM T16688 C02SPM 71771026 IC50 = 94 nM T16688 C2HQB0 71771027 IC50 = 170 nM T16688 C1SY2B 71771028 IC50 = 50 nM T16688 CNB4T6 71771029 IC50 = 79 nM T16688 C8PHX5 71771030 IC50 = 174 nM T16688 C6B3JF 71812428 IC50 > 10000 nM T16688 C92NTY 71812429 IC50 > 10000 nM T16688 C1TY7V 71812430 IC50 > 10000 nM T16688 C41WTO 71812431 IC50 > 10000 nM T16688 CDI59F 71812432 IC50 = 330 nM T16688 CA2M0F 71812620 IC50 > 10000 nM T16688 CWQU40 71812621 IC50 > 10000 nM T16688 CSN7I6 71812622 IC50 = 90 nM T16688 C5JV1P 71812623 IC50 = 112 nM T16688 C0IJ9V 71812624 IC50 = 49 nM T16688 C35OXS 71812811 IC50 > 10000 nM T16688 C5FRX9 71812812 IC50 > 10000 nM T16688 CAPI35 71812813 IC50 = 1070 nM T16688 CNOB18 71812814 IC50 = 2010 nM T16688 CIMR74 71815039 IC50 > 10000 nM T16688 C67SJQ 71815040 IC50 > 10000 nM T16688 C2E3UH 72164408 IC50 = 1.7 nM T16688 CE19XB 72164409 IC50 = 2 nM T16688 CIQ14A 72164530 IC50 = 5.3 nM T16688 CW82TS 72164531 IC50 = 1.3 nM T16688 CQX62C 72164657 IC50 = 3.2 nM T16688 CJB5H4 72164658 IC50 = 772 nM T16688 C5LMZ3 72164659 IC50 = 101 nM T16688 C4G7HK 72164774 IC50 = 32 nM T16688 CJ8WK2 72164775 IC50 = 11 nM T16688 CDI29X 72188386 IC50 = 120 nM T16688 C2NPJ4 72188424 IC50 = 83 nM T16688 CO6CE2 72188428 IC50 = 540 nM T16688 CBT10U 72188430 IC50 = 390 nM T16688 CI2L0B 72545068 IC50 = 1712 nM T16688 CK04HO 72545069 IC50 = 1616 nM T16688 CF6YM8 72545070 IC50 = 1560 nM T16688 CC0J7N 72545071 IC50 = 2837 nM T16688 CRCA61 72545307 IC50 = 84 nM T16688 CY7X0I 72545308 IC50 = 179 nM T16688 CB32SL 72545309 IC50 = 116 nM T16688 C7H6RK 72545310 IC50 = 103 nM T16688 CL3XM9 73345986 IC50 = 16 nM T16688 C5FT1H 73345987 IC50 = 20 nM T16688 C7GK2C 73346029 IC50 = 1060 nM T16688 C3CL9P 73347519 IC50 = 23 nM T16688 CNZ84J 73349048 IC50 = 10 nM T16688 C04XEI 73349049 IC50 = 49 nM T16688 CHO2Y9 73352119 IC50 = 22 nM T16688 C1H5RN 73352120 IC50 = 58 nM T16688 CS2KE3 73355079 IC50 = 82 nM T16688 C48QWV 73355080 IC50 = 97 nM T16688 CU5E0J 73356638 IC50 = 23 nM T16688 CPZ5T6 73356639 IC50 = 37 nM T16688 CV81GS 73356640 IC50 = 101 nM T16688 C2P6ZX 76311188 IC50 = 8 nM T16688 CM14WO 76318402 IC50 = 199.53 nM T16688 C85FJM 76322077 IC50 = 1258.93 nM T16688 C3F1IY 76332913 IC50 = 140 nM T16688 C2T1RX 76332914 IC50 = 794.33 nM T16688 CQ9H4U 86277844 IC50 = 64 nM T16688 CI21JL 86765197 IC50 = 14.8 nM T16688 C71QCV 89582842 IC50 = 1.6 nM T16688 CC94YO 89584863 IC50 = 2.1 nM T16688 CNZ2I8 89584875 IC50 = 5.2 nM T16688 CIBL54 89584906 IC50 = 1.3 nM T16688 CQY4J1 89584935 IC50 = 1.7 nM T16688 C9FCS1 90644592 IC50 = 43 nM T16688 CSKY85 90644593 IC50 = 32 nM T16688 CH9OM3 90644594 IC50 = 91 nM T16688 C7TP1X 90644595 IC50 = 85 nM T16688 CQ15NV 90644596 IC50 = 230 nM T16688 CR2PH0 90644597 IC50 = 290 nM T16688 C6BQ4E 90644598 IC50 = 530 nM T16688 CGFS97 90644599 IC50 = 580 nM T16688 C8H0KU 90644600 IC50 = 580 nM T16688 CKD4T2 90644601 IC50 = 3700 nM T16688 C4JCK7 90644602 IC50 = 140 nM T16688 CTO70U 90654628 IC50 > 10000 nM T16688 CBIG20 90654629 IC50 > 10000 nM T16688 CXFY30 90654929 IC50 = 72.85 nM T16688 C49PWF 90654930 IC50 = 75.59 nM T16688 C1HR0A 90654931 IC50 = 34.15 nM T16688 C86LCQ 90654932 IC50 = 149.9 nM T16688 C1IK2P 90654933 IC50 = 20.4 nM T16688 CUE5C4 90654934 IC50 = 38.88 nM T16688 C5H3RF 90654935 IC50 = 26.2 nM T16688 CX9WK2 90654936 IC50 = 54.85 nM T16688 C6OBI1 90655566 IC50 = 36 nM T16688 CJ4Z7M 90655567 IC50 = 448 nM T16688 CCY26G 90655568 IC50 = 58 nM T16688 CO0J5U 90655569 IC50 = 122 nM T16688 CF27IH 90668345 IC50 = 31.62 nM T16688 CA6R4G 90668346 IC50 = 5.012 nM T16688 C0B5RL 90668347 IC50 = 316.23 nM T16688 COZ97H 90668348 IC50 = 15.85 nM T16688 CO0T3D 90668349 IC50 = 79.43 nM T16688 CQE37T 90668350 IC50 = 31.62 nM T16688 CU98TM 118467765 IC50 = 126 nM T16688 C41DNT 118467787 IC50 = 158 nM T16688 C2RBF7 118918048 IC50 > 10000 nM T16688 CSBO65 122179027 IC50 > 30000 nM T16688 C6KCR0 122188918 IC50 = 539 nM T16688 C19NIE 122188919 IC50 > 50000 nM T16688 CLC27I 122188920 IC50 = 201 nM T16688 CYBD82 122188921 IC50 > 50000 nM T16688 C65PKO 122188922 IC50 > 50000 nM T16688 C70CKQ 122188923 IC50 = 34 nM T16688 C75SHP 122188924 IC50 = 5 nM T16688 CDUP05 122188925 IC50 = 89 nM T16688 CK0I4A 122188926 IC50 > 10000 nM T16688 CF61HK 122188927 IC50 > 500 nM T16688 CW40LZ 122188928 IC50 = 159 nM T16688 CMS89O 122188929 IC50 > 10000 nM T16688 CZ4R7S 122188930 IC50 > 10000 nM T16688 CY82ZE 122188931 IC50 = 32 nM T16688 CRS2J0 122188932 IC50 > 500 nM T16688 CZL5W4 122188933 IC50 > 500 nM T16688 CW6GU3 122188934 IC50 = 300 nM T16688 C62TDW 122188935 IC50 = 105 nM T16688 CEUL85 122188936 IC50 = 280 nM T16688 CJOC12 122188937 IC50 = 170 nM T16688 C8HN7U 122189249 IC50 = 31000 nM T16688 CNV03S 122189255 IC50 > 50000 nM T16688 CKT6V0 123320121 IC50 = 70 nM T16688 CA94XD 123818187 IC50 = 65 nM T16688 C7AK4V 127028635 IC50 = 7 nM T16688 C2BPX8 127028636 IC50 = 11 nM T16688 CIB1M6 127028637 IC50 = 27 nM T16688 C2VY1L 127028638 IC50 > 10000 nM T16688 CN1R3D 127028952 IC50 > 10000 nM T16688 C7BK9P 127028953 IC50 = 4800 nM T16688 CB03UV 127028954 IC50 = 3500 nM T16688 CTF8Q1 127028955 IC50 = 1400 nM T16688 CRBZ04 127028956 IC50 = 760 nM T16688 CV7A4J 127028957 IC50 = 62 nM T16688 C8UX4Q 127034759 IC50 > 10000 nM T16688 C3PSV1 127042393 IC50 = 3 nM T16688 C5QCS7 135979913 IC50 = 570 nM T16688 C3E0VL 136046112 IC50 = 7900 nM T16688 C5KI7Q 136264975 IC50 = 451 nM T16688 C6B5US 137628648 IC50 = 3 nM T16688 CTB0D5 137631556 IC50 = 364 nM T16688 C7IL8G 137631604 IC50 > 10000 nM T16688 CR7ZC3 137632040 IC50 = 1642 nM T16688 CBGO67 137633268 IC50 = 3775 nM T16688 CJQ9C2 137634281 IC50 = 102 nM T16688 CH45GD 137635354 IC50 = 4249 nM T16688 CJYH94 137635550 IC50 = 643 nM T16688 C6UW0T 137639828 IC50 = 29 nM T16688 CM8QN6 137640037 IC50 = 6584 nM T16688 CCI1P6 137640495 IC50 = 62 nM T16688 CH38MC 137640679 IC50 = 36 nM T16688 CUOT01 137640920 IC50 = 7036 nM T16688 CW53GX 137641132 IC50 = 95 nM T16688 CX4HU2 137641521 IC50 = 207 nM T16688 C9EMH2 137641995 IC50 = 29 nM T16688 CAY2I5 137645058 IC50 = 2957 nM T16688 C02USX 137645633 IC50 = 25 nM T16688 CT8F1Z 137647286 IC50 = 5136 nM T16688 CHI20J 137649152 IC50 = 697 nM T16688 C7V1IB 137649471 IC50 = 37.7 nM T16688 C57SOY 137649945 IC50 = 6 nM T16688 C0WUA3 137652176 IC50 = 2200 nM T16688 C8N9IR 137652534 IC50 = 8704 nM T16688 C76QHP 137653064 IC50 = 89 nM T16688 CRVG50 137653102 IC50 = 151 nM T16688 C26FMT 137653184 IC50 = 74 nM T16688 CPW2X3 137653563 IC50 = 131 nM T16688 C29PSM 137654796 IC50 = 7543 nM T16688 CR1TG3 137655891 IC50 = 966 nM T16688 CZ4W3T 137656391 IC50 > 10000 nM T16688 CRKM68 137657957 IC50 = 1407 nM T16688 C5T9GK 137662102 IC50 = 216 nM T16688 CB40JN 145949401 IC50 = 8 nM T16688 C6YZJ1 145951921 IC50 = 8 nM T16688 CV53YE 145958014 IC50 = 3 nM T16688 CTHA94 145958032 IC50 = 20 nM T16688 C4ORE1 145960378 IC50 = 21 nM T16688 C5B4XG 145960732 IC50 = 1929 nM T16688 CS61CL 145960927 IC50 = 35 nM T16688 C4MN1K 145961350 IC50 = 5502 nM T16688 CF1G2E 145961610 IC50 = 14 nM T16688 CY7F8B 145961755 IC50 = 1241 nM T16688 CB24EW 145962028 IC50 = 468 nM T16688 C9L5JB 145962193 IC50 = 55 nM T16688 CXLA86 145962260 IC50 = 387 nM T16688 C42PLT 145962320 EC50 = 26 nM T16688 C8T9RL 145962381 IC50 = 429 nM T16688 CSP5J1 145962746 IC50 = 44 nM T16688 C1WXU2 145962877 IC50 = 74 nM T16688 CQM0C4 145962913 IC50 = 281 nM T16688 C0MQH7 145962966 IC50 = 210 nM T16688 C03YDQ 145963005 IC50 = 25 nM T16688 CM9U1Z 145963257 IC50 = 120 nM T16688 C2Q1HN 145963285 IC50 = 15 nM T16688 CLP89H 145963384 EC50 = 20 nM T16688 CJX28D 145963431 IC50 = 94 nM T16688 C56HJV 145963462 IC50 = 30 nM T16688 CJ5VR4 145979853 IC50 = 100 nM T16688 C4MQU9 145980134 IC50 > 50000 nM T16688 CH62PL 145986440 IC50 = 199.53 nM T16688 C87YAI 145989147 IC50 = 100 nM T16688 CLN9U5 145990619 IC50 = 39.81 nM T16688 C6GQV8 145992185 IC50 = 125.89 nM T16688 CM9JE5 145992670 IC50 = 50.12 nM T16688 C48PKI 155511086 IC50 = 41 nM T16688 CM1BV9 155523387 IC50 = 22 nM T16688 CH06BN 155523388 IC50 = 66 nM T16688 CT4B0F 155527719 IC50 = 1.7 nM T16688 CT1JB7 155528212 IC50 = 5.4 nM T16688 CHR60D 155528366 IC50 = 8 nM T16688 CN7I6O 155528434 IC50 = 3.1 nM T16688 C4L7ZO 155530653 IC50 = 4.1 nM T16688 C7UBH8 155532385 IC50 = 3.5 nM T16688 C85MAE 155537732 IC50 = 12600 nM T16688 CSMI71 155540479 IC50 = 2.4 nM T16688 CST86Y 155544326 IC50 = 5.3 nM T16688 CD9KW4 155544699 IC50 = 3.6 nM T16688 CI92YC 155546800 IC50 = 2.9 nM T16688 C9I1SL 155550029 IC50 = 150 nM T16688 C6F8YA 155555651 IC50 = 9 nM T16688 C8PI6V 155556175 IC50 = 4.2 nM T16688 D02RUZ 24768261 IC50 = 7 nM T16555 CP5SG4 448872 EC50 = 567 nM T16555 C0GYD6 448923 EC50 = 2500 nM T16555 CU4CS9 11146048 EC50 = 562 nM T16555 CHB3C7 11510273 Ki = 3300 nM T16555 CT74ZJ 11560464 Ki > 15000 nM T16555 CUD1J5 11611428 Ki = 5950 nM T16555 CAP5Z8 16220801 EC50 = 880 nM T16555 CO7FT9 16220889 EC50 = 11 nM T16555 C9V8KY 16221095 EC50 = 1880 nM T16555 CIX4T8 22838429 EC50 = 320 nM T16555 C5M6KP 24858471 EC50 = 361 nM T16555 CI3D1T 44422868 EC50 > 10000 nM T16555 CQW7S1 44422870 EC50 = 49 nM T16555 CWQ57Y 44422899 EC50 = 420 nM T16555 CH57TE 44440209 EC50 = 370 nM T16555 C3QST4 44440213 EC50 = 810 nM T16555 CA2U7V 44585948 EC50 = 63 nM T16555 CT01NA 44627485 EC50 = 4580 nM T16555 CYP17B 44627487 EC50 = 0.92 nM T16555 CL3D1N 44627489 EC50 = 2730 nM T16555 CACW71 44627490 EC50 = 56 nM T16555 CM1R2N 44627590 EC50 = 39 nM T16555 CN8U1Z 44627592 EC50 = 40 nM T16555 CGX9A2 44627594 EC50 = 7460 nM T16555 CM3IS5 44627596 EC50 = 480 nM T16555 CHB4D5 44627598 EC50 = 11 nM T16555 CD35BV 44627689 EC50 = 1600 nM T16555 CR4CO5 44627691 EC50 = 167 nM T16555 C7BHI9 44627693 EC50 = 252 nM T16555 CE6XH9 44627695 EC50 = 32 nM T16555 CQKW67 44627697 EC50 = 5160 nM T16555 CT32KD 44627698 EC50 = 5160000 nM T16555 CQ2V9E 44627699 EC50 = 768 nM T16555 CGT23C 44627801 EC50 = 1490 nM T16555 C5P2FB 44627803 EC50 = 1800 nM T16555 C51QDF 44627805 EC50 = 1900 nM T16555 CF6XN5 45485237 EC50 = 142 nM T16555 C12QZE 45485253 EC50 = 3320 nM T16555 CV6US7 46226441 EC50 = 588 nM T16555 CH1C7V 46226445 EC50 = 2590 nM T16555 CB7NY5 46226446 EC50 = 496 nM T16555 CVJ31P 46226447 EC50 = 323 nM T16555 C9RTX3 46226448 EC50 = 1880 nM T16555 CB8C1P 46226454 EC50 = 373 nM T16555 CM8TW4 46226455 EC50 = 905 nM T16555 CPR7F4 46226456 EC50 = 658 nM T16555 C16QVJ 46226460 EC50 = 238 nM T16555 CO71DL 46226463 EC50 = 951 nM T16555 C8CK9F 46226477 EC50 = 460 nM T16555 CI65GM 46890713 EC50 = 140 nM T16555 C1WXL6 49861324 EC50 = 3320 nM T16555 CSHG53 54584734 EC50 = 671 nM T16555 C4VFI2 68530100 Ki = 2350 nM T16555 CM75YG 122185397 IC50 = 362 nM T16555 C52AMG 124221651 Ki = 0.08 nM T16555 CL7U5X 126720243 IC50 = 5690 nM T16555 CM57GR 126720252 IC50 = 25.4 nM T16555 CA56TL 132280527 IC50 = 31.7 nM T16555 CGN13V 134611895 IC50 = 169 nM T16555 CK9UA8 135356790 IC50 = 228 nM T16555 C31RPN 135356798 IC50 = 224 nM T16555 C8M4GA 135356877 IC50 = 162 nM T16555 C21TCP 135356879 IC50 = 481 nM T16555 CGI08F 135356919 IC50 = 72.4 nM T16555 C60YGL 135356965 IC50 = 237 nM T16555 CZT63Y 135357071 IC50 = 115 nM T16555 C6WGT5 135357363 IC50 = 290 nM T16555 C0H6DS 135357364 IC50 = 91 nM T16555 C4RG1U 139392057 IC50 = 763 nM T16555 CJ1UO6 145964206 IC50 = 566 nM T16555 C32LBA 145964225 IC50 = 8420 nM T16555 CT4FW3 145964454 IC50 = 33100 nM T16555 C2L8BR 145965191 IC50 = 13600 nM T16555 CLS09A 145965286 IC50 = 756 nM T16555 C4WFL8 145965747 IC50 = 2280 nM T16555 CF4L9T 145965887 IC50 = 2260 nM T16555 CCY9H7 145966012 IC50 = 899 nM T16555 C2MS3R 145966170 IC50 = 269 nM T16555 CM7YH1 145966357 IC50 = 3110 nM T16555 CT9UQ0 145966524 IC50 = 6440 nM T16555 C5ZBN8 145966901 IC50 = 516 nM T16555 CAFL85 145966990 IC50 = 1190 nM T16555 CA70RS 145968000 IC50 = 1510 nM T16555 CC7Y2T 145969364 IC50 = 563 nM T16555 C8L9RV 145969418 IC50 = 83.5 nM T16555 CHB42F 145969817 IC50 = 1410 nM T16555 CGB6U5 145970281 IC50 = 2430 nM T16555 C7BYR5 145971306 IC50 = 9330 nM T16555 CN7QX1 145971541 IC50 = 12600 nM T16555 CB2WA9 145972038 IC50 = 608 nM T16555 C29NDC 145972815 IC50 = 1490 nM T16555 CT5CX0 145973771 IC50 = 133 nM T16555 CM3PX6 145974515 IC50 = 26800 nM T16555 CJ8RK4 145974993 IC50 = 1640 nM T16555 CTQ96O 145975403 IC50 > 50000 nM T16555 CHGD31 145975592 IC50 = 2180 nM T16555 C8IHX5 145976578 IC50 = 5920 nM T16555 CC9OI4 145977136 IC50 = 1750 nM T16555 CJUO19 145977176 IC50 = 735 nM T16555 C38MVJ 145977351 IC50 = 53000 nM T16555 C8IEY0 145977566 IC50 = 16400 nM T16555 CEAK62 145977711 IC50 = 7530 nM T16555 CPQ09I 145977780 IC50 = 1960 nM T16555 CMKX43 145977870 IC50 = 67200 nM T16555 C86HTC 145977897 IC50 = 958 nM T16555 C36ITN 145978183 IC50 = 54700 nM T16555 CDE7Z5 145978299 IC50 = 3200 nM T16555 C5M7ZS 145978515 IC50 = 10900 nM T16555 CXI26C 145978641 IC50 = 20700 nM T16555 C2QH5U 155512121 IC50 = 1.77 nM T16555 C5LUP8 155516521 IC50 > 3000 nM T16555 CS9P0C 155525228 IC50 = 4.54 nM T16555 C9OH6Q 155525420 IC50 = 131 nM T16555 C5XL4A 155526332 IC50 = 4.95 nM T16555 CT83QU 155540535 IC50 = 6660 nM T16555 C6QRM5 155544120 IC50 = 5.06 nM T16555 C8ZR7Q 155549217 IC50 = 4.35 nM T16555 CP02KU 155564566 IC50 = 3.17 nM T16555 D02HAL 6031 EC50 = 160 nM T16555 D03WBX 44585949 EC50 = 11 nM T16555 D05MXI 42611190 IC50 = 0.4 nM T16555 D07MIE 8629 EC50 = 261 nM T16555 D07MTB 11510579 Ki = 3500 nM T16555 D07TSE 16082712 EC50 = 1.92 nM T16555 D0K7WW 18068 EC50 = 670 nM T16555 D0O8AN 17473 EC50 = 370 nM T16555 D0Z9JO 448873 EC50 = 910 nM T82309 D0B2WJ 3371 EC50 > 100000 nM T82309 D0X4RN 3676 IC50 > 100000 nM T82309 C0D4UM 11594207 EC50 = 45000 nM T82309 CFS98J 16078951 EC50 = 6000 nM T82309 C6MCY1 134151176 EC50 = 18800 nM T34389 CB9GM4 176443 Ki = 1200 nM T34389 CMJ30V 5353845 Ki = 80 nM T34389 CY6D5H 9821458 Ki = 2.3 nM T34389 CZ10UR 9905153 Ki = 11 nM T34389 CHT5U3 10044204 Ki = 7.8 nM T34389 CAV1F0 10066884 IC50 = 0.11 nM T34389 C0I5WV 10453439 IC50 ~ 10000 nM T34389 CI68UO 11393923 Ki = 7.5 nM T34389 CU94ZT 11484453 Ki = 0.29 nM T34389 C4JB6X 11587811 Ki = 850 nM T34389 CG2B7X 11631387 Ki = 1 nM T34389 C0QJ9O 11652690 Ki = 0.85 nM T34389 C57KVO 11674428 Ki = 1 nM T34389 CG7O5E 11695972 Ki = 0.77 nM T34389 CV74JA 11696246 Ki = 0.83 nM T34389 CAG6H2 11709766 Ki = 2000 nM T34389 C8G9AL 16756850 IC50 = 6300 nM T34389 C3D7RI 18530647 IC50 > 1000 nM T34389 C1IQ9L 22486206 Ki = 0.39 nM T34389 C0PE9N 25021166 IC50 = 5410 nM T34389 C4OVH1 25021168 IC50 = 2660 nM T34389 C4KRB0 44201123 IC50 = 9 nM T34389 CS59IP 44340580 IC50 = 2 nM T34389 C8RTA7 44389776 Ki = 0.52 nM T34389 CS1JH5 44389963 Ki = 16 nM T34389 CGA87C 44389967 Ki = 0.29 nM T34389 C84ISX 44389973 Ki = 3 nM T34389 CJ91NL 44391726 Ki = 0.56 nM T34389 CSP9G2 44396041 IC50 = 37400 nM T34389 C4DL5C 44469677 IC50 = 8 nM T34389 CTK1R9 44478601 IC50 = 220 nM T34389 C4PNA1 44479144 IC50 > 1000 nM T34389 C65YHX 44479149 IC50 > 1000 nM T34389 CCZF08 44479896 IC50 = 10 nM T34389 CF2VN0 44482522 IC50 = 69 nM T34389 C6XIR9 44482524 IC50 = 760 nM T34389 CT40WX 44482525 IC50 = 401 nM T34389 C62GOP 44563661 IC50 = 42 nM T34389 CLOM59 44563664 IC50 = 0.15 nM T34389 C0S7GK 45103520 IC50 = 5 nM T34389 C36IAE 45103521 IC50 > 100000 nM T34389 CO5PY9 45104436 IC50 > 50000 nM T34389 CM6U2I 45104437 IC50 = 4340 nM T34389 C8ZL3I 45104438 IC50 = 3500 nM T34389 CN0F3J 45104535 IC50 = 5850 nM T34389 CF2VT8 45104537 IC50 = 40080 nM T34389 CBG20U 45104539 IC50 = 9000 nM T34389 CVS1N3 45104540 IC50 > 50000 nM T34389 C5BF6A 45104639 IC50 > 50000 nM T34389 CZA1W7 45104759 IC50 = 5830 nM T34389 C3NJ9L 45104760 IC50 = 15100 nM T34389 CRIS48 45104761 IC50 > 50000 nM T34389 C4PAQ0 45104762 IC50 = 10540 nM T34389 C6E4VZ 45104856 IC50 = 3360 nM T34389 CHZ25L 45104857 IC50 = 4690 nM T34389 CWD6Z4 45104859 IC50 = 380 nM T34389 CM6PE1 45104860 IC50 = 1040 nM T34389 CKOJ29 45104954 IC50 = 1050 nM T34389 CJ76GA 45104955 IC50 = 4600 nM T34389 C4D0VY 45104956 IC50 = 3570 nM T34389 CL29IY 45104957 IC50 = 930 nM T34389 CH1S8N 45104958 IC50 = 40 nM T34389 CEN4I6 45104959 IC50 = 280 nM T34389 C3D2HJ 45105055 IC50 = 20 nM T34389 C6I4MX 45105056 IC50 = 720 nM T34389 CMI7T1 45105057 IC50 = 5 nM T34389 CI71OZ 45105058 IC50 = 40 nM T34389 CBH8V9 45105059 IC50 = 40 nM T34389 CZK3J7 45105060 IC50 = 90 nM T34389 C0HZ4C 46916514 Ki = 0.18 nM T34389 C93OCD 46916515 Ki = 60 nM T34389 CBL01G 46916516 Ki = 4.8 nM T34389 CFL18K 46916517 Ki = 32 nM T34389 C3SIH7 46916518 Ki = 140 nM T34389 CDBM59 46916519 Ki = 0.49 nM T34389 CW6Y2D 46916520 Ki = 0.5 nM T34389 CDRP69 46916562 IC50 > 200 nM T34389 C6CH7R 46916564 IC50 > 70 nM T34389 CCDO74 46916565 IC50 > 200 nM T34389 CTK84W 46916566 IC50 > 70 nM T34389 CX0PM9 46916567 IC50 > 200 nM T34389 CRZ52S 49862864 IC50 > 50000 nM T34389 CG2O4F 49862865 IC50 = 200 nM T34389 C5S0TV 49862894 IC50 > 50000 nM T34389 CZ8ME2 49862911 IC50 = 17 nM T34389 CXB26I 49862912 IC50 = 28 nM T34389 C21TML 49862913 IC50 = 232 nM T34389 CS9TI3 49862914 IC50 = 100 nM T34389 CE7P5Q 49862938 IC50 > 50000 nM T34389 CB8AU5 49862939 IC50 = 116 nM T34389 CA0ZO1 49862940 IC50 = 112 nM T34389 CXVZ46 49862941 IC50 = 84 nM T34389 CQ34VU 49862971 IC50 > 25000 nM T34389 C6YS4V 56679834 IC50 = 12 nM T34389 CU70JQ 60199625 Ki = 8 nM T34389 C3LU4X 60199626 Ki = 18 nM T34389 CX0T5E 60199627 Ki = 7 nM T34389 C6KC9M 60199628 Ki = 11 nM T34389 C5QIL0 60201942 IC50 > 10000 nM T34389 CB1RN0 60201943 IC50 > 50000 nM T34389 CK0Q7M 60201944 IC50 > 200 nM T34389 C91BHF 60202099 IC50 > 200 nM T34389 C7WT4J 60202100 IC50 > 200 nM T34389 CPQ4B5 60202101 IC50 > 50000 nM T34389 CYUN89 60202102 IC50 > 200 nM T34389 C8X5ZV 60202103 IC50 > 200 nM T34389 CY96BG 60202104 Ki = 23 nM T34389 CXSA80 66671848 Ki = 0.16 nM T34389 C6T9BL 71533603 Ki = 10 nM T34389 CZ3X6K 71533604 Ki = 13 nM T34389 C67QMT 71540959 Ki = 270 nM T34389 CI8R4P 71540960 Ki = 263 nM T34389 CRL40K 71540961 Ki > 500 nM T34389 C30PXT 71541069 Ki > 500 nM T34389 CB5AR0 71541070 Ki > 500 nM T34389 CE8N4X 71541071 Ki = 240 nM T34389 C6YRN2 71541072 Ki > 500 nM T34389 CL9V0F 71541073 Ki > 500 nM T34389 CT2ER7 71541074 Ki > 500 nM T34389 CQ9D6U 71665477 IC50 = 30 nM T34389 C7BY9P 71665478 IC50 < 10 nM T34389 C68QPX 76325440 IC50 < 10 nM T34389 C76KWI 76332658 IC50 < 10 nM T34389 CV4FI5 76336259 IC50 = 80 nM T34389 CM10KY 76336262 IC50 = 270 nM T34389 CEU20D 85470198 Ki = 3000 nM T34389 C4ZQJ7 89785475 IC50 = 2200 nM T34389 C1WIX6 89847041 IC50 = 1000 nM T34389 CX79VN 90656092 IC50 = 50 nM T34389 C8E6JX 90656103 IC50 = 90 nM T34389 CH0K8Y 90656104 IC50 = 460 nM T34389 CX1T5J 92135986 IC50 < 10 nM T34389 CZ9T6H 118526557 IC50 < 10 nM T34389 CX3VW5 118526625 IC50 = 60 nM T34389 C2N7BP 118526627 IC50 = 650 nM T34389 CEV5P6 118526739 IC50 = 960 nM T34389 C4E7HU 118526750 IC50 < 10 nM T34389 CURN41 118526755 IC50 = 90 nM T34389 CO6HG9 118526928 IC50 < 10 nM T34389 CJGL98 118526975 IC50 = 560 nM T34389 C3DP0R 118709041 IC50 = 800 nM T34389 C03GXE 118709042 IC50 = 1200 nM T34389 CBR1K9 118709043 IC50 = 60 nM T34389 C1ZP4G 130431469 IC50 = 350 nM T34389 CMA35H 130431481 IC50 = 510 nM T34389 CT89XU 145951627 Ki = 6300 nM T34389 C5IA9S 145977816 IC50 = 12 nM T34389 CQ46AJ 155513119 IC50 = 790000 nM T34389 CBRT63 155518073 IC50 > 100000 nM T34389 CR8Q7L 155518672 Ki = 420 nM T34389 C83EJB 155520173 IC50 > 1000000 nM T34389 CO45NM 155520675 Ki = 50 nM T34389 CJ4K7U 155525568 IC50 > 100000 nM T34389 C6G2ZH 155525932 IC50 > 1000000 nM T34389 C61VMW 155527042 IC50 = 8700 nM T34389 C1AP0Z 155527970 IC50 > 100000 nM T34389 C1P4DY 155529475 IC50 = 3000 nM T34389 CSD83T 155531974 IC50 > 100000 nM T34389 C71YMQ 155535169 Ki = 0.23 nM T34389 CDL9R5 155536374 Ki = 16 nM T34389 C8WRH2 155540919 Ki = 203 nM T34389 CQN3I9 155541938 Ki = 194 nM T34389 C50AMQ 155542534 Ki = 46 nM T34389 CE5I1R 155544612 IC50 = 120 nM T34389 C3UFK5 155547686 IC50 > 100000 nM T34389 C0DHX7 155550192 Ki = 16 nM T34389 CX7YR1 155551280 IC50 = 190 nM T34389 CPXZ31 155555424 IC50 = 510 nM T34389 C76IMR 155555589 Ki = 25 nM T34389 C4YT7O 155556111 IC50 = 450 nM T34389 CEA7D4 155557420 IC50 > 100000 nM T34389 C1U4ZL 155560181 Ki = 6.88 nM T34389 C9AK3H 155561632 IC50 = 9000 nM T34389 CNR68T 155561836 IC50 > 100000 nM T34389 CMV43N 155564327 IC50 > 1000000 nM T34389 C0PD3V 155567316 IC50 > 100000 nM T34389 D00QUN 44563663 IC50 = 3 nM T34389 D00ULT 10609180 Ki = 130 nM T34389 D02ENI 10293363 Ki = 370 nM T34389 D02JVI 44387731 Ki = 220 nM T34389 D03ZBS 44563662 IC50 = 12 nM T34389 D04PMA 15353606 Ki = 140 nM T34389 D04YUA 162019 IC50 = 1.9 nM T34389 D06MNW 44285344 Ki = 100 nM T34389 D06UDN 46232606 IC50 = 13 nM T34389 D07GOA 11150976 Ki = 0.28 nM T34389 D08XQI 9395 IC50 = 540 nM T34389 D08YHD 9878121 Ki = 170 nM T34389 D09GVB 10427006 Ki = 4.7 nM T34389 D0B1BQ 157730 Ki = 240 nM T34389 D0CH0K 11327355 Ki = 18 nM T34389 D0D0FX 44389962 Ki = 90 nM T34389 D0G0MZ 25021165 IC50 = 4000 nM T34389 D0H6FG 10429254 IC50 = 0.1 nM T34389 D0HQ4M 24762154 IC50 = 3 nM T34389 D0K6GY 49864679 IC50 = 0.4 nM T34389 D0M7SQ 9795477 Ki = 25 nM T34389 D0M8AR 11154099 Ki = 320 nM T34389 D0N1CK 9813810 Ki = 100 nM T34389 D0NH1E 1383884 Ki = 1.2 nM T34389 D0OJ7E 35027739 IC50 = 14 nM T34389 D0R5RW 45104861 IC50 = 930 nM T34389 D0T4HB 44563660 IC50 = 0.1 nM T34389 D0TN0A 10085812 Ki = 0.2 nM T34389 D0U0CV 18516661 IC50 = 2 nM T34389 D0W6PT 21804 IC50 = 40 nM T34389 D0W7XR 11507802 IC50 = 12.4 nM T01280 D00XKB 57406537 Ki = 7.5 nM T01280 D04OSA 46202416 IC50 = 0.9 nM T01280 D0N1BF 44251605 IC50 = 2880 nM T01280 D0O8UB 53241828 IC50 = 24 nM T01280 D0R4KK 51352361 IC50 = 0.38 nM T01280 D0Y0EP 67979346 IC50 = 0.9 nM T01280 D0Y5NA 118435360 IC50 = 194 nM T01280 D0H4IY 59262421 Ki = 7.8 nM T01280 CXU5P7 213731 IC50 = 87190 nM T01280 C8NGY9 448772 IC50 = 137000 nM T01280 CGSC72 5287532 IC50 = 132 nM T01280 CRS54N 6540293 Ki = 356 nM T01280 CLF04H 9938431 IC50 = 96 nM T01280 CW67YS 9939419 IC50 = 170 nM T01280 C2P3DU 9983140 IC50 = 5010 nM T01280 CIBZ30 9984485 IC50 > 10 nM T01280 C93KNF 9986236 IC50 = 8320 nM T01280 CHG57R 9986500 IC50 = 10110 nM T01280 C8XV3Y 10008157 IC50 = 4485 nM T01280 CN2J9E 10054920 IC50 = 420 nM T01280 CY9SK0 10073810 IC50 = 41690 nM T01280 CEFK38 10077756 IC50 = 4215 nM T01280 CAKR94 10077830 IC50 = 435 nM T01280 CJ4TR1 10078059 IC50 = 160 nM T01280 CSA7C0 10098656 IC50 = 3243 nM T01280 C0LOV8 10100288 IC50 = 870 nM T01280 CK51FX 10100482 IC50 = 620 nM T01280 CC2I7B 10212352 IC50 = 500 nM T01280 C2UNQ0 10258545 IC50 = 3615 nM T01280 CB60PQ 10258985 IC50 = 430 nM T01280 CJZ98B 10324013 IC50 = 3610 nM T01280 C3QN7I 10326962 IC50 = 580 nM T01280 CM46XO 10327211 IC50 = 42 nM T01280 CML3K5 10348155 IC50 = 7590 nM T01280 CN89XA 10369729 IC50 = 44670 nM T01280 CQ0Y7C 10371570 IC50 = 580 nM T01280 CIA94Y 10371854 IC50 = 510 nM T01280 CZ5J7R 10391277 IC50 = 63100 nM T01280 CZK1G9 10413386 IC50 = 12020 nM T01280 CYL37G 10415909 IC50 = 2000 nM T01280 CEYO32 10416248 IC50 = 655 nM T01280 C8F3EC 10438938 IC50 = 6920 nM T01280 CJU80M 10439665 IC50 = 145 nM T01280 CZ6GK9 10461757 IC50 = 765 nM T01280 CYE70D 10483879 IC50 = 780 nM T01280 C74JHX 10483887 IC50 = 480 nM T01280 CN68BR 10484078 IC50 = 24550 nM T01280 C3RQ9I 11157167 IC50 = 590 nM T01280 C6HBJ0 11168125 IC50 = 3100 nM T01280 CEX8G1 11178891 IC50 = 1170 nM T01280 C06BES 11192316 IC50 = 75 nM T01280 CN8IX6 11215318 IC50 = 1047 nM T01280 CY7IP9 11215540 IC50 = 114 nM T01280 COWF09 11215541 IC50 = 210 nM T01280 CJHM10 11227304 IC50 = 89 nM T01280 CH81IQ 11227430 IC50 = 390 nM T01280 CU0C8V 11238286 IC50 = 370 nM T01280 CG87MJ 11250223 IC50 = 620 nM T01280 CU80VL 11290116 IC50 > 50000 nM T01280 C9E0FG 11295146 IC50 = 1490 nM T01280 C4WK2S 11295726 IC50 = 1140 nM T01280 C7FKT1 11296858 IC50 = 59 nM T01280 CNS4B0 11296859 IC50 = 59 nM T01280 CM3G0J 11308211 IC50 = 210 nM T01280 CY5GU3 11308212 IC50 = 110 nM T01280 CVDC34 11329962 IC50 = 430 nM T01280 CL0P2H 11342148 IC50 = 420 nM T01280 C2LFN6 11342476 IC50 = 360 nM T01280 C5QL8O 11376341 IC50 = 443 nM T01280 CY78LG 11377351 IC50 = 680 nM T01280 CHX8E5 11410816 IC50 = 69 nM T01280 CIPA26 11410903 IC50 = 110 nM T01280 C84MEW 11421906 IC50 = 260 nM T01280 CEM8Q5 11444313 IC50 = 263 nM T01280 C3ZI7O 11444912 IC50 = 150 nM T01280 CR4F1K 11456236 IC50 = 3020 nM T01280 CLK8V9 11467715 IC50 = 350 nM T01280 C0OPF5 11467778 IC50 = 940 nM T01280 CH2Y7V 11478322 IC50 = 2170 nM T01280 C7LAQ1 11493476 IC50 = 24400 nM T01280 CRZ86I 11498384 Ki = 458 nM T01280 C2LD3N 11510567 IC50 = 170 nM T01280 CK0L9W 11510740 IC50 = 16700 nM T01280 C3P6ZU 11516577 IC50 = 780 nM T01280 CYIV63 11517020 IC50 = 2800 nM T01280 CW68BJ 11518143 IC50 > 30000 nM T01280 C5XB3T 11520033 IC50 = 51 nM T01280 C2VN5E 11531131 IC50 = 540 nM T01280 CIK75C 11532248 IC50 = 1000 nM T01280 CPK79W 11532880 IC50 = 3600 nM T01280 C2W8MQ 11538592 IC50 = 960 nM T01280 CT50OI 11539235 IC50 = 1840 nM T01280 C6CVW2 11539562 IC50 = 7540 nM T01280 CR93VK 11539712 IC50 = 10700 nM T01280 C2IL9N 11543843 IC50 = 38300 nM T01280 CS8MV6 11544960 IC50 = 30100 nM T01280 C0KY4O 11545958 IC50 = 560 nM T01280 CYEL51 11553053 IC50 = 7000 nM T01280 CSL71C 11553983 IC50 = 960 nM T01280 CE9ZI8 11556254 IC50 = 45 nM T01280 CZ07VP 11560610 IC50 = 2320 nM T01280 C5UR7S 11578047 IC50 = 20 nM T01280 CE6CH3 11583947 IC50 = 2300 nM T01280 CA29QF 11589453 IC50 = 4170 nM T01280 CZ1V8Y 11606008 IC50 = 500 nM T01280 C92XGC 11609507 Ki = 139 nM T01280 CT97EJ 11611402 IC50 = 600 nM T01280 C1PSL5 11614083 IC50 = 54 nM T01280 CFU9Q3 11618427 IC50 = 22400 nM T01280 C7ZWK0 11620576 IC50 = 470 nM T01280 C9R6UV 11624078 Ki = 30 nM T01280 CUD76B 11632510 IC50 = 520 nM T01280 C78KYL 11633041 IC50 = 6600 nM T01280 C2QC4B 11633904 IC50 = 300 nM T01280 COC2F0 11639859 IC50 = 550 nM T01280 CED2Y7 11640634 IC50 = 3500 nM T01280 C8DZG9 11647909 IC50 = 3780 nM T01280 C6MH7K 11648455 IC50 = 11400 nM T01280 C0UXN3 11654224 IC50 = 500 nM T01280 CSKL32 11654876 IC50 = 200 nM T01280 C4PXM5 11668120 IC50 = 1130 nM T01280 C14JYI 11668187 IC50 = 1590 nM T01280 C4G6YQ 11684817 IC50 = 1000 nM T01280 C7SPG0 11692473 IC50 = 620 nM T01280 CK73DU 11710655 IC50 = 10900 nM T01280 CBJ08S 11711024 IC50 = 16180 nM T01280 C7ZRM9 11719190 IC50 = 7100 nM T01280 CF1CZ0 11765081 IC50 = 690 nM T01280 CN7AX1 11765192 IC50 = 68 nM T01280 CJN0K9 11765311 IC50 = 1510 nM T01280 CF1RT6 11785879 IC50 = 1260 nM T01280 CG2HY0 11785880 IC50 = 1260 nM T01280 CVQ7O2 11786748 IC50 = 210 nM T01280 CLP92O 11963435 IC50 > 30000 nM T01280 CGOD35 11990754 IC50 = 120 nM T01280 CQ8SJ5 11990755 IC50 = 2370 nM T01280 CR4G6J 15949919 IC50 = 190 nM T01280 CQ3GX2 15950003 IC50 = 50 nM T01280 C3CI9Z 15950004 IC50 = 50 nM T01280 C2BQ4V 15950005 IC50 = 130 nM T01280 C6QD9U 15950006 IC50 = 150 nM T01280 CW4US1 15950085 IC50 = 8790 nM T01280 CZM1C9 15950086 IC50 = 870 nM T01280 C8Y6UT 15950518 IC50 = 190 nM T01280 CAPV27 15950520 IC50 = 570 nM T01280 C20LCO 15950595 IC50 = 1170 nM T01280 C6DCB3 15950597 IC50 = 1020 nM T01280 C49WLN 15950662 IC50 = 24100 nM T01280 CK4L8W 15950666 IC50 = 480 nM T01280 C0OCS6 15950667 IC50 = 2200 nM T01280 C3WIC9 15951413 IC50 = 2010 nM T01280 C0J9PD 15951416 IC50 = 140 nM T01280 CSQ3X1 15951420 IC50 = 80 nM T01280 C8IZR0 15951484 IC50 = 60 nM T01280 CB1G7D 15951486 IC50 = 140 nM T01280 CNPJ39 15951487 IC50 = 40 nM T01280 C2XJU6 15951488 IC50 = 1010 nM T01280 CE67NK 15951489 IC50 = 20 nM T01280 CW6S0H 15981486 IC50 = 177 nM T01280 C0QAD8 16050550 IC50 = 680 nM T01280 C1CEU6 16050551 IC50 = 2530 nM T01280 CX8O6Q 16050552 IC50 = 5550 nM T01280 CYQ7X3 16050553 IC50 = 4330 nM T01280 C2WR8B 16050640 IC50 = 830 nM T01280 CF5EC0 16050641 IC50 = 9590 nM T01280 CN0F8Z 16050834 IC50 = 410 nM T01280 CD5W4A 16050837 IC50 = 1650 nM T01280 C4DO8C 16050931 IC50 = 510 nM T01280 C8R6HZ 16050932 IC50 = 170 nM T01280 C21JUT 16050937 IC50 = 120 nM T01280 C72ZAL 16050938 IC50 = 310 nM T01280 CL35CA 16051038 IC50 = 570 nM T01280 C2CJ4S 16051040 IC50 = 270 nM T01280 CQCJ80 16051495 IC50 = 490 nM T01280 CRAS90 16051584 IC50 = 1850 nM T01280 C0Q2MC 16051586 IC50 = 30 nM T01280 CW6CX4 16051696 IC50 = 180 nM T01280 CL4I9N 16051697 IC50 = 40 nM T01280 CE3L1D 16051698 IC50 = 20 nM T01280 CAY1B5 16090342 IC50 = 12900 nM T01280 CP5G7V 16090348 IC50 = 340 nM T01280 C2HMT5 16113206 IC50 = 280 nM T01280 CX39UL 16113753 IC50 = 1300 nM T01280 CL26VD 16659019 Ki = 556 nM T01280 CU62LO 16659020 Ki = 523 nM T01280 CGU76F 16659022 Ki = 408 nM T01280 C73FHN 16659067 Ki = 340 nM T01280 C01GFZ 16659107 Ki = 397 nM T01280 CRW5Q2 16730753 IC50 = 12 nM T01280 CK40YS 23657802 IC50 = 5890 nM T01280 C4BR2E 23657804 IC50 = 3600 nM T01280 CEI3N7 24794397 IC50 = 1160 nM T01280 CJUX10 24808497 IC50 = 22 nM T01280 CWM1Q4 24878892 IC50 = 32360 nM T01280 CTO0H5 24878893 IC50 = 32360 nM T01280 CKWX57 24878894 IC50 = 7940 nM T01280 CF0Q3S 24878945 IC50 = 19500 nM T01280 C09LYN 24878946 IC50 = 19500 nM T01280 CI54AT 24878947 IC50 = 47860 nM T01280 C8LQ5C 24882338 IC50 = 1810 nM T01280 CMJK34 24882477 IC50 = 370 nM T01280 C32SYP 24950594 IC50 = 2000 nM T01280 CO7MQ2 25069561 IC50 = 370 nM T01280 C8ANG7 25070193 IC50 = 160 nM T01280 C0T8LP 25070195 IC50 = 850 nM T01280 CM37LQ 25072736 IC50 = 50 nM T01280 C0UO6V 25073049 IC50 = 110 nM T01280 CMYC57 25115954 IC50 = 21 nM T01280 CNTF43 25127621 IC50 = 70 nM T01280 C4E0MJ 25127622 IC50 = 120 nM T01280 CWF5Z3 25143506 IC50 > 30000 nM T01280 CP89ZX 25181420 IC50 > 100000 nM T01280 C4JQ0L 25181421 IC50 > 100000 nM T01280 C3XDW1 25184934 IC50 = 10800 nM T01280 CS2MU5 25184935 IC50 = 17300 nM T01280 CXE56W 25184936 IC50 = 7300 nM T01280 CF91ST 25184937 IC50 = 12200 nM T01280 CSM9C5 25190481 IC50 = 26840 nM T01280 CU80RW 25190482 IC50 = 4130 nM T01280 CK48PJ 25190483 IC50 = 3080 nM T01280 CW6QJ1 25190484 IC50 = 1050 nM T01280 CKZ2Q7 25190485 IC50 = 4680 nM T01280 CWN51E 25190486 IC50 = 1020 nM T01280 C69RHT 25190487 IC50 = 1450 nM T01280 CT8N2P 25190488 IC50 = 1660 nM T01280 CJ6SA2 25190489 IC50 = 760 nM T01280 CESB62 25190490 IC50 = 600 nM T01280 CLS3O2 25190491 IC50 = 2290 nM T01280 CZY6C4 25190492 IC50 = 2950 nM T01280 C04QGB 25190493 IC50 = 6920 nM T01280 CF8U0N 25190494 IC50 = 4270 nM T01280 CX4PB5 25190495 IC50 = 630 nM T01280 CKYP06 25190496 IC50 = 13215 nM T01280 CNXG37 25190497 IC50 > 100000 nM T01280 CTS92Q 25190499 IC50 = 785 nM T01280 CY02QR 25190500 IC50 = 2465 nM T01280 CXV1A7 44143258 IC50 = 9120 nM T01280 CWI68J 44143259 IC50 = 8130 nM T01280 CNQ97G 44143260 IC50 = 7080 nM T01280 C95LPG 44143261 IC50 = 4170 nM T01280 CV9K7F 44143262 IC50 = 5750 nM T01280 C0WRT2 44143263 IC50 = 8320 nM T01280 CWQ6L4 44143264 IC50 = 5750 nM T01280 CZ9MQ7 44143265 IC50 = 6310 nM T01280 C8EI0C 44143266 IC50 = 8910 nM T01280 CAJ0I2 44143267 IC50 = 5130 nM T01280 C7AH8B 44143268 IC50 = 12590 nM T01280 CFJ82W 44143269 IC50 = 13180 nM T01280 CQ34LK 44143270 IC50 = 23440 nM T01280 C7FQ8W 44143271 IC50 = 350 nM T01280 CCUX36 44143272 IC50 = 7760 nM T01280 CDR56H 44143274 IC50 = 3590 nM T01280 CNWC13 44143275 IC50 = 11190 nM T01280 C4C0WD 44143276 IC50 = 18710 nM T01280 C5SLK9 44143277 IC50 = 28 nM T01280 C39WZR 44143278 IC50 = 1230 nM T01280 CVF5L8 44143280 IC50 = 13550 nM T01280 CPX9B2 44143282 IC50 = 331 nM T01280 C6CQM2 44143283 IC50 = 260 nM T01280 CDEU24 44143285 IC50 = 3200 nM T01280 CD8WS6 44143286 IC50 = 1150 nM T01280 CJ8DS1 44198935 IC50 = 10.2 nM T01280 CXC57A 44421346 IC50 = 230 nM T01280 CA71VT 44421347 IC50 = 210 nM T01280 CU4B2Y 44441701 IC50 = 1600 nM T01280 C6QMY7 44441703 IC50 = 54000 nM T01280 C2JE8M 44441743 IC50 = 41000 nM T01280 C68VFD 44446196 IC50 = 42000 nM T01280 C4S1CA 44446197 IC50 = 12020 nM T01280 C7K1RZ 44446198 IC50 = 5890 nM T01280 C5CS2Z 44446199 IC50 = 57540 nM T01280 CZO7A4 44446200 IC50 = 3090 nM T01280 CJVG08 44446201 IC50 = 30200 nM T01280 CF7RP8 44446202 IC50 = 69010 nM T01280 CU54SK 44446203 IC50 = 600 nM T01280 CJ3BD7 44446204 IC50 = 21380 nM T01280 CJW16S 44446205 IC50 = 3390 nM T01280 CSPE84 44446206 IC50 = 3720 nM T01280 CS42CJ 44446207 IC50 = 93330 nM T01280 C7VX1Q 44446209 IC50 = 15140 nM T01280 CG4N8T 44446210 IC50 = 6920 nM T01280 C1HZ9O 44446211 IC50 = 33100 nM T01280 CN2AB7 44446212 IC50 = 33110 nM T01280 CH6G1V 44447299 IC50 > 100000 nM T01280 CXS7Y3 44454508 IC50 = 5130 nM T01280 C2QI1J 44454509 IC50 = 28600 nM T01280 CML29V 44454541 IC50 = 78530 nM T01280 CBS73X 44454542 IC50 > 100000 nM T01280 CJ0NI6 44454543 IC50 > 21000 nM T01280 C0XMF7 44454839 IC50 = 1580 nM T01280 CTY3G5 44454842 IC50 = 8793 nM T01280 CIFD60 44454874 IC50 = 830 nM T01280 CP08GW 44454875 IC50 = 650 nM T01280 CU9GD7 44454913 IC50 = 12880 nM T01280 C6XY2B 44454914 IC50 = 8235 nM T01280 C7OGW4 44454944 IC50 = 4790 nM T01280 C10PVS 44454945 IC50 = 400 nM T01280 C9SB5E 44455462 IC50 = 4000 nM T01280 CI7GZ9 44455467 IC50 = 2600 nM T01280 C24BWX 44455486 IC50 = 2400 nM T01280 CZSO57 44455487 IC50 = 4250 nM T01280 C5A7CY 44455514 IC50 = 330 nM T01280 CEKI49 44455515 IC50 = 260 nM T01280 CY68NV 44455516 IC50 = 1200 nM T01280 CLT1R8 44455543 IC50 = 400 nM T01280 CL9N0S 44455544 IC50 = 6200 nM T01280 CJ3V2W 44455567 IC50 = 1350 nM T01280 CI34FJ 44455570 IC50 = 1070 nM T01280 CS2HG8 44455573 IC50 = 5600 nM T01280 CGW49Q 44455601 IC50 = 1400 nM T01280 CD7GY0 44455602 IC50 = 3600 nM T01280 CN3JK0 44455638 IC50 = 2130 nM T01280 C1VD5W 44455639 IC50 = 2150 nM T01280 CAQ03Z 44455666 IC50 = 5150 nM T01280 CQFW59 44455691 IC50 = 1500 nM T01280 C2A6DO 44455692 IC50 = 1700 nM T01280 CS16QI 44455695 IC50 = 1200 nM T01280 C5HQN3 44455724 IC50 = 2000 nM T01280 CGK5A1 44455750 IC50 = 795 nM T01280 CT8QL3 44455753 IC50 = 582 nM T01280 CU0NA7 44455754 IC50 = 1200 nM T01280 C3X7BU 44455772 IC50 = 610 nM T01280 CJ4I3V 44455775 IC50 = 2300 nM T01280 CH8IB5 44455802 IC50 = 5000 nM T01280 CAGM05 44478390 IC50 = 10500 nM T01280 C9P3XR 44478656 IC50 = 9900 nM T01280 CJ7AL5 44478659 IC50 = 4400 nM T01280 CCO70V 44570172 IC50 > 100000 nM T01280 CMNO27 44570173 IC50 > 100000 nM T01280 C26UXD 44570174 IC50 > 100000 nM T01280 C9JI2N 44570207 IC50 > 100000 nM T01280 C0CFU7 44570208 IC50 > 100000 nM T01280 CCN7P9 44570209 IC50 > 100000 nM T01280 CL8SM0 44570210 IC50 > 100000 nM T01280 CVW7F2 44570211 IC50 = 141 nM T01280 C34VYL 44570212 IC50 = 251 nM T01280 C78FBX 44570213 IC50 > 100000 nM T01280 CSE6U7 44570261 IC50 = 2089 nM T01280 COI30F 44570262 IC50 = 1949 nM T01280 CJ2MR9 44570263 IC50 > 100000 nM T01280 CTB4F0 44570302 IC50 > 100000 nM T01280 C1Q0DR 44570303 IC50 > 100000 nM T01280 CQ9G6O 44631933 IC50 = 810 nM T01280 C3M7ZG 45105274 Ki = 5.4 nM T01280 C2YE7A 45254510 IC50 = 5 nM T01280 CK76PW 45255111 IC50 = 85 nM T01280 C43HDC 45256109 IC50 = 15 nM T01280 C8BYZ2 45259044 IC50 = 370 nM T01280 CIY5X1 45267880 IC50 = 1860 nM T01280 CD2MC1 45268670 IC50 = 450 nM T01280 C16WVK 45269615 IC50 = 5460 nM T01280 C4NTM7 45488098 IC50 = 230 nM T01280 C6W8LK 45488101 IC50 = 3870 nM T01280 CHMZ65 45488102 IC50 = 6290 nM T01280 C4GVA9 45488103 IC50 = 5160 nM T01280 CT51JC 45488104 IC50 = 4020 nM T01280 C1Q9DK 45488105 IC50 = 1640 nM T01280 CJ13RL 45488106 IC50 = 9970 nM T01280 CH7SG2 45488107 IC50 = 1260 nM T01280 CL0H9O 45488108 IC50 = 73580 nM T01280 C9KP7N 45488109 IC50 = 1190 nM T01280 CJ75VZ 45488110 IC50 = 5040 nM T01280 C4QV8Z 45488111 IC50 = 2480 nM T01280 C4ZD5W 45488112 IC50 = 5990 nM T01280 CXG2R1 45488113 IC50 = 420 nM T01280 C9NG1H 45488114 IC50 = 1720 nM T01280 C8FTJ3 45488115 IC50 = 1840 nM T01280 CB10OE 45488116 IC50 = 2510 nM T01280 CE1ZX5 45488119 IC50 = 780 nM T01280 CKBT31 45488120 IC50 = 9690 nM T01280 CH0W9R 45488121 IC50 = 1840 nM T01280 C38LWQ 46202743 Ki = 1700 nM T01280 CNVX45 46205968 Ki = 790 nM T01280 C3VYC6 46217866 IC50 = 170 nM T01280 CH2EI5 46218828 Ki = 120 nM T01280 CY9O4P 46225190 IC50 = 510 nM T01280 CQMD65 46225238 IC50 = 490 nM T01280 CZS8H2 46225290 IC50 = 1150 nM T01280 C4O6GY 46231497 IC50 = 6130 nM T01280 C1K6QJ 46231500 IC50 = 23600 nM T01280 C8THA6 46231554 IC50 = 11000 nM T01280 CK3O2Q 46231555 IC50 = 6700 nM T01280 CZK5E9 46238536 IC50 = 8000 nM T01280 C6KN1D 46830239 IC50 = 100 nM T01280 CNP2S7 46844428 IC50 = 140 nM T01280 C7D4SK 46844429 IC50 = 200 nM T01280 CO5QC2 46881646 IC50 = 1500 nM T01280 C7C2EK 46881691 IC50 = 3800 nM T01280 CWB9C6 46881692 IC50 = 3700 nM T01280 CJN4Y2 46881693 IC50 = 960 nM T01280 CS0O9T 46883935 IC50 = 130 nM T01280 CDO30L 46883936 IC50 = 700 nM T01280 C7O3XP 46884002 IC50 = 1000 nM T01280 CHT53N 49797544 IC50 = 1430 nM T01280 CD4W0Y 49797545 IC50 = 4370 nM T01280 CI8FT3 49836033 IC50 = 840 nM T01280 CR41SW 49863021 IC50 = 600 nM T01280 C9O7UP 49863022 IC50 = 8900 nM T01280 C9OWG2 49863023 IC50 = 7100 nM T01280 CNC25U 49863024 IC50 = 4100 nM T01280 CED4S9 49863025 IC50 = 79400 nM T01280 CCY4G0 49863026 IC50 = 132000 nM T01280 C8T0LZ 49863027 IC50 = 35000 nM T01280 CSYU53 49863028 IC50 = 46000 nM T01280 C64OTC 49863029 IC50 = 117000 nM T01280 CWP2N9 49863030 IC50 = 200000 nM T01280 CWK1B5 49863031 IC50 = 1260 nM T01280 C19EDA 49869312 IC50 = 110 nM T01280 CD62TH 49869313 IC50 = 30 nM T01280 CO3CN1 50898731 IC50 = 602 nM T01280 CD64NT 51039270 IC50 = 3.3 nM T01280 CJ6M8H 52940810 IC50 = 350 nM T01280 C3DN8M 52940827 IC50 = 120 nM T01280 CVT4K3 52940915 IC50 = 2680 nM T01280 CLJ01Q 52942108 IC50 = 500 nM T01280 CX16LC 52942291 IC50 = 11700 nM T01280 CHN91J 52942848 IC50 = 210 nM T01280 CQPD40 52944421 IC50 = 140 nM T01280 CQ4V8R 52946545 IC50 = 730 nM T01280 CRIQ87 52946950 IC50 = 2480 nM T01280 CWC0D6 52946966 IC50 = 2830 nM T01280 CB3NQ0 52948140 IC50 = 400 nM T01280 CY34UI 52948154 IC50 = 320 nM T01280 CKT0J6 52948174 IC50 = 100 nM T01280 C2XIY3 52949466 IC50 = 170 nM T01280 CPO5A7 52950127 IC50 = 40 nM T01280 C2D1JV 53230332 IC50 = 10 nM T01280 C32QSO 53240812 IC50 = 9440 nM T01280 C6V5GK 53241151 IC50 = 52 nM T01280 C17AMV 53241205 IC50 = 106 nM T01280 CLZC60 53241206 IC50 = 18 nM T01280 CDQJ08 53241302 IC50 = 11 nM T01280 CA9EF1 53241709 IC50 = 15 nM T01280 CC86WU 53241710 IC50 = 22 nM T01280 CR2AW3 53241825 IC50 = 12 nM T01280 C0BRK7 53241826 IC50 = 36 nM T01280 CZ56VB 53241932 IC50 = 23 nM T01280 C7H1ZP 53241933 IC50 = 7490 nM T01280 C2F8QG 53241937 IC50 = 31 nM T01280 C17GML 53465141 IC50 = 0.8 nM T01280 CF40KI 54580003 IC50 = 28180 nM T01280 CG1D6V 56658432 IC50 = 450 nM T01280 C0RMT9 56658435 IC50 = 20 nM T01280 C2J7TS 56658436 IC50 = 680 nM T01280 CW8IY4 56658437 IC50 = 1150 nM T01280 C45YJU 56658717 IC50 = 20 nM T01280 CS4MX1 56658718 IC50 = 30 nM T01280 CM4P2G 56661917 IC50 = 500 nM T01280 C4QD7Z 56661918 IC50 = 620 nM T01280 C47HVP 56661919 IC50 = 230 nM T01280 CQP28A 56665390 IC50 = 120 nM T01280 C39XJR 56668818 IC50 = 7390 nM T01280 CXW4B7 56668819 IC50 = 36 nM T01280 C1Z7MG 56668820 IC50 = 560 nM T01280 C10MSR 56668821 IC50 = 50 nM T01280 C5VIR4 56669107 IC50 = 6650 nM T01280 C1DFQ6 56672294 IC50 = 170 nM T01280 CFE52J 56672296 IC50 = 650 nM T01280 C2EZ8O 56672297 IC50 = 3120 nM T01280 CGNH26 56672298 IC50 = 70 nM T01280 CCG59L 56672299 IC50 = 410 nM T01280 CLP36K 56672300 IC50 = 20 nM T01280 C43PXS 56675689 IC50 = 210 nM T01280 CL8PK3 56675694 IC50 = 490 nM T01280 CV3BE8 56675695 IC50 = 440 nM T01280 CUI46G 56675696 IC50 = 70 nM T01280 CO7G3P 56678998 IC50 = 18 nM T01280 C65LKQ 56678999 IC50 = 610 nM T01280 CLW2C5 56679000 IC50 = 740 nM T01280 CH80FW 56679262 IC50 = 860 nM T01280 CGL67Z 56682312 IC50 = 20 nM T01280 C07EXO 56682313 IC50 = 780 nM T01280 CE8PW7 56682314 IC50 = 5450 nM T01280 C7QB6A 56682567 IC50 = 1470 nM T01280 CBVK48 56834873 Ki = 3568 nM T01280 C7SIV2 56834949 IC50 = 29 nM T01280 C4KP9I 56925448 Ki = 5509 nM T01280 C0ZKP8 56925449 Ki = 3617 nM T01280 CQE1L7 56925450 Ki = 2810 nM T01280 C9DH8A 56925452 Ki = 3674 nM T01280 CMSO49 56925453 Ki = 4110 nM T01280 CG3C2H 56925544 Ki = 4003 nM T01280 CE9YN7 56925547 Ki = 3777 nM T01280 C92CRT 56925548 Ki = 3081 nM T01280 CNV7I5 56925549 Ki = 3224 nM T01280 CO3BA4 57390575 Ki = 2281 nM T01280 CQ58OT 57395865 Ki = 1733 nM T01280 CVJZ32 57395866 Ki = 1818 nM T01280 C0YAU9 57399319 Ki = 2354 nM T01280 CVL27Z 57399320 Ki = 2065 nM T01280 C8NEZ3 57401086 Ki = 2067 nM T01280 CWCY97 57406911 Ki = 740 nM T01280 C2K9PU 59250417 IC50 = 316 nM T01280 CCS34R 59250998 IC50 = 10 nM T01280 CJ54VX 59262314 Ki = 170 nM T01280 CS8KD6 59262423 Ki = 360 nM T01280 COXS29 59262510 Ki = 68 nM T01280 C2PJ4N 59271992 IC50 > 30000 nM T01280 CJKM47 59374702 IC50 = 14 nM T01280 C85IUE 59387407 Ki = 11 nM T01280 CQW7A8 60149247 Ki = 480 nM T01280 C60ESV 60194610 IC50 = 26.3 nM T01280 CFML30 66665322 IC50 = 6 nM T01280 C56CFA 68448803 IC50 > 10000 nM T01280 CG5MW2 71273898 IC50 = 4 nM T01280 CE69IS 71273947 IC50 = 580 nM T01280 CQD14Z 71274016 IC50 = 71 nM T01280 CY5NV8 71274019 IC50 = 71 nM T01280 CES40A 71305034 IC50 = 904 nM T01280 CEV0B7 71449561 IC50 = 3.9 nM T01280 C92RIS 71449970 Ki = 78 nM T01280 C86RHK 71451365 IC50 > 10000 nM T01280 CL7P2A 71451832 Ki = 770 nM T01280 C2NM4Q 71455471 Ki = 1450 nM T01280 CLG93R 71459108 Ki = 11 nM T01280 CV0E9B 71460380 IC50 = 4.5 nM T01280 CBO2M4 71460381 IC50 = 390 nM T01280 C6OC0Z 71460382 IC50 = 88 nM T01280 CP6IV2 71462074 IC50 = 22 nM T01280 CD4QU0 71462075 IC50 = 1900 nM T01280 C0GBL7 71466345 IC50 = 86.3 nM T01280 C2Z6UE 71468021 Ki = 17.4 nM T01280 C1FL6A 71529262 IC50 = 290 nM T01280 C10UQB 71529265 IC50 = 2900 nM T01280 CB8DU6 71529426 IC50 = 7 nM T01280 CBO09H 71529465 IC50 = 66 nM T01280 CU8QX2 71582923 IC50 = 245900 nM T01280 CLS5E7 71582924 IC50 = 319000 nM T01280 CUB68J 71583022 IC50 > 1000000 nM T01280 C0B1QM 71584523 IC50 > 1000000 nM T01280 C1NP5F 71584646 IC50 = 207200 nM T01280 CXO41P 71584647 IC50 = 193800 nM T01280 C63BJM 71584648 IC50 = 100500 nM T01280 C6S0IQ 71584649 IC50 = 21000 nM T01280 CGET05 71584650 IC50 = 33200 nM T01280 CIGV69 71619629 IC50 = 101 nM T01280 CV7G9C 71663691 IC50 = 30 nM T01280 CX73JM 71663692 IC50 = 47 nM T01280 CQ57VI 71663693 IC50 = 45 nM T01280 CE4DJ8 71663694 IC50 = 245 nM T01280 C9UN3Q 71663695 IC50 = 119 nM T01280 C1H2BL 71663858 IC50 = 943 nM T01280 C54DZH 71714118 IC50 = 1340 nM T01280 CP56WO 71718352 IC50 = 175 nM T01280 C5DC0Z 72946535 IC50 = 4300 nM T01280 C8K6NI 72946537 IC50 = 5700 nM T01280 CQM8U4 72946738 IC50 = 10100 nM T01280 CQ3DV8 72946943 IC50 = 4400 nM T01280 CYXC78 72947373 IC50 = 8900 nM T01280 CLYH10 75593331 Ki = 1 nM T01280 C0X1HW 85470889 Ki = 1 nM T01280 C8EK2Y 85471653 Ki = 1.2 nM T01280 CC2T7G 86291837 IC50 = 19.5 nM T01280 C5XON4 86293009 IC50 = 19.05 nM T01280 CZLX91 86294744 IC50 = 5.3 nM T01280 C7OIC6 86762648 IC50 = 295 nM T01280 CVD2I6 88602735 IC50 = 30 nM T01280 C4GAU0 90656187 IC50 = 4550 nM T01280 CB1C5A 90656190 IC50 = 25.12 nM T01280 CAQ05V 90693645 Ki = 71 nM T01280 CWZX73 91971958 IC50 = 7.1 nM T01280 CLP6K8 117960375 Ki = 9 nM T01280 C74EMN 118190070 Ki = 17 nM T01280 C94WRZ 118435363 IC50 = 3.9 nM T01280 C1WL4E 118435382 IC50 = 367 nM T01280 C5L9VH 118435403 IC50 = 60.7 nM T01280 CNXH97 118435407 IC50 = 20 nM T01280 C8Z2FP 118435412 IC50 = 233 nM T01280 CJIP45 118435414 IC50 = 1072 nM T01280 CY6EP7 118435506 IC50 = 1709 nM T01280 CPE35X 118435524 IC50 = 57 nM T01280 CVK6Y8 118435560 IC50 = 338 nM T01280 C37SFM 118435617 IC50 = 38.9 nM T01280 CL6IV1 118440826 IC50 = 44.1 nM T01280 CHIL17 118441142 IC50 = 72.3 nM T01280 C5W2NL 118865901 IC50 = 0.8 nM T01280 C5NE9P 118866030 IC50 < 2 nM T01280 COR8Y4 118866094 IC50 = 1.8 nM T01280 CELZ36 118866105 IC50 = 18.6 nM T01280 C9Z1BW 118866133 IC50 = 31 nM T01280 CWCX50 118866162 IC50 = 562 nM T01280 CZ7SF8 118866177 IC50 = 34 nM T01280 C2CZ5B 118866257 IC50 = 12 nM T01280 CK2U6X 118866347 IC50 < 2 nM T01280 CQ5Y3R 118866403 IC50 = 94 nM T01280 C4MLU1 118866454 IC50 < 2 nM T01280 CH6AT4 118866474 IC50 < 2 nM T01280 CA51SU 118866499 IC50 = 39.4 nM T01280 C68ELY 118866551 IC50 = 40 nM T01280 CGIC35 118866737 IC50 = 401 nM T01280 CM2N6G 118866838 IC50 < 2 nM T01280 CIM4Y6 118866963 IC50 < 2 nM T01280 C9M2WU 118866986 IC50 = 9.7 nM T01280 CT4Z2R 118884907 IC50 = 1.1 nM T01280 CX8JW2 118885049 IC50 = 40 nM T01280 CP13NA 118958876 Ki = 3 nM T01280 CFW1D5 118974304 Ki = 207.2 nM T01280 CRW25M 121264059 Ki = 14 nM T01280 CGH84P 121264098 Ki = 303 nM T01280 C2XA0P 121298035 IC50 = 141.25 nM T01280 CO7E4P 122180108 IC50 = 497 nM T01280 CJM51V 122180111 IC50 = 22700 nM T01280 C15DUY 122180113 IC50 = 584 nM T01280 C13ELK 122180115 IC50 = 26300 nM T01280 CXMQ41 122180117 IC50 = 11100 nM T01280 CZ5VM7 122180628 Ki = 7.3 nM T01280 CKFA52 122180629 Ki = 14.2 nM T01280 CSN78D 122180630 Ki = 18.3 nM T01280 C05VYD 122180631 Ki = 12.7 nM T01280 C2R6SY 122197438 IC50 = 16220 nM T01280 CDG6R0 122197443 IC50 = 3800 nM T01280 CG8H6M 122435134 Ki = 3.5 nM T01280 CIFT47 122484483 IC50 = 479 nM T01280 C35XVL 122535397 Ki = 51 nM T01280 CGLX79 122653795 IC50 = 17.6 nM T01280 CK7W8B 123132907 IC50 = 405 nM T01280 CRW0C2 123132915 IC50 = 228 nM T01280 C45OVL 126693206 IC50 = 29.9 nM T01280 C1E7IG 126693231 IC50 = 129 nM T01280 CUF68P 126961340 Ki = 7140 nM T01280 CIK56O 129201653 Ki = 16 nM T01280 C4IQ6F 129201655 Ki = 3 nM T01280 CH5V3A 129201660 Ki = 1 nM T01280 C5Q1GT 129202050 Ki = 6 nM T01280 C19KGT 129202057 Ki = 1 nM T01280 CCBV68 129202062 Ki = 1 nM T01280 C7H3QJ 129202063 Ki = 1 nM T01280 CVMY58 129202069 Ki = 3 nM T01280 CLH8Z9 129202106 Ki = 6 nM T01280 CV78UP 132054712 Ki = 2022 nM T01280 CO63CX 132054802 Ki = 21 nM T01280 CX27OU 132054828 Ki = 1299 nM T01280 CRJA89 132054902 Ki = 2077 nM T01280 C4UH5R 132054950 Ki = 443 nM T01280 CD7AZ2 132068809 Ki = 13 nM T01280 CXR7J9 132604796 IC50 = 120 nM T01280 CMA13L 134284187 IC50 = 446 nM T01280 C9W6JQ 135125856 IC50 = 51 nM T01280 CKVF19 135126469 IC50 = 52 nM T01280 CI1D7K 135875806 IC50 = 1500 nM T01280 CV0Y1W 136266507 Ki = 10.9 nM T01280 CES5F6 137462330 Ki = 3.4 nM T01280 C8JWF7 137633017 IC50 = 27300 nM T01280 CU40QT 137634377 IC50 = 1010 nM T01280 CLK7A3 137635011 IC50 = 7130 nM T01280 CY5M8Z 137635828 IC50 = 62900 nM T01280 C2B1MZ 137637375 IC50 = 35900 nM T01280 CEVA49 137637780 IC50 = 75700 nM T01280 CXG42C 137638912 Ki = 817 nM T01280 CSQL63 137640486 IC50 > 100000 nM T01280 CKC6N9 137641085 Ki = 1478 nM T01280 C91GMY 137641491 IC50 > 100000 nM T01280 C9BF0V 137643369 IC50 = 7600 nM T01280 CV56QL 137645221 IC50 = 1890 nM T01280 CG3U5K 137645264 Ki = 134 nM T01280 C9OV2Q 137646113 Ki = 13 nM T01280 CTB27V 137646126 IC50 = 19400 nM T01280 C10CBD 137646316 IC50 > 100000 nM T01280 CLF8P5 137646591 Ki = 1011 nM T01280 CJXK40 137648425 IC50 > 94000 nM T01280 CVR29E 137651451 IC50 = 11500 nM T01280 C8HSX7 137652983 IC50 = 26800 nM T01280 CL3DW0 137653017 Ki = 710 nM T01280 CQ32NO 137653545 IC50 = 1020 nM T01280 CBE82Q 137653962 Ki = 2193 nM T01280 CXY7F1 137654633 IC50 > 100000 nM T01280 CTU5C1 137656577 IC50 = 17500 nM T01280 C3L8WX 137657646 IC50 > 84000 nM T01280 C1ULD3 137660988 Ki = 13 nM T01280 C3YFL4 137662127 IC50 > 100000 nM T01280 C1MRT7 138454796 Ki = 1740 nM T01280 C8DH9F 138857908 IC50 = 28 nM T01280 CE35GB 138857909 IC50 = 13 nM T01280 C48XFW 142342111 IC50 = 14.5 nM T01280 C45TMN 145960757 Ki = 198 nM T01280 C1KMU8 145961539 Ki = 0.5 nM T01280 COI9X0 145962778 Ki = 9 nM T01280 CVU70C 145962834 Ki = 10 nM T01280 CYTQ79 153303564 IC50 = 170 nM T01280 CBC6S2 154031826 IC50 = 6.607 nM T01280 C83RXG 154031827 IC50 = 79.43 nM T01280 CM7U1J 155513259 IC50 = 37.15 nM T01280 CL53YZ 155513311 IC50 = 0.19 nM T01280 C7V8ZP 155516667 IC50 = 1660 nM T01280 CU9B6X 155517833 IC50 = 1 nM T01280 CSU3P7 155518836 IC50 = 26.92 nM T01280 C1H7YT 155520705 IC50 = 3.02 nM T01280 CKO59Y 155522051 IC50 = 251 nM T01280 C40DMT 155526564 Ki = 1 nM T01280 CUY0L8 155528391 IC50 = 13.2 nM T01280 COW05C 155536534 Ki = 1 nM T01280 CKGP95 155536618 IC50 = 56.23 nM T01280 COF63Z 155537873 IC50 = 0.5 nM T01280 CUK21B 155538074 IC50 < 2 nM T01280 C2B5ID 155538495 Ki = 14 nM T01280 C1W7DO 155538806 IC50 = 15.8 nM T01280 C4TQN1 155542315 IC50 = 43.65 nM T01280 CB9V1D 155543145 Ki = 32 nM T01280 CF6XZ8 155544727 IC50 = 16.6 nM T01280 CPHJ28 155548834 IC50 = 275.42 nM T01280 CQ2J3F 155556725 IC50 = 66 nM T01280 CLYI80 155559529 IC50 = 102 nM T01280 C2KUE9 155560600 IC50 = 78 nM T01280 C7BCO6 155563658 IC50 = 94 nM T01280 CBS97E 155565975 Ki = 479 nM T01280 C93SNX 155566643 IC50 = 74 nM T01280 C0QJL4 155568510 IC50 = 602 nM T01280 D00SDQ 50938551 IC50 = 9 nM T01280 D02LCH 16659106 Ki = 31 nM T01280 D04RSC 447068 Ki = 3 nM T01280 D07EWF 66575082 Ki < 1 nM T01280 D08ALW 449218 Ki = 4.5 nM T01280 D09SOY 15054176 IC50 = 770 nM T15556 D0JI2E 10224267 IC50 = 8600 nM T15556 D02QBJ 6450819 IC50 = 2700 nM T15556 D0YK7C 9932718 IC50 = 3500 nM T15556 CA7BM2 4271052 IC50 = 50000 nM T15556 CA7ZE2 6505361 IC50 = 51000 nM T15556 CM06PH 9797139 IC50 = 59400 nM T15556 CY0Q9R 9810857 IC50 = 590 nM T15556 CUX19E 9829598 IC50 = 200 nM T15556 CULH64 9832101 IC50 = 220 nM T15556 CMS65P 9832433 IC50 = 10700 nM T15556 CTQX65 9853548 IC50 = 2480 nM T15556 C5IHC1 9854049 IC50 = 140 nM T15556 CN4WI2 9869327 IC50 = 10 nM T15556 CRG7Q3 9875505 IC50 = 130 nM T15556 C5CHU0 9875587 IC50 = 480 nM T15556 C7J9TI 9895968 IC50 = 100 nM T15556 CGHO67 9897158 IC50 = 6060 nM T15556 C43FBS 9918721 IC50 = 2280 nM T15556 CFLD01 9937280 IC50 = 1400 nM T15556 CLJ6N7 9940247 IC50 = 2400 nM T15556 C9R4XL 9940626 IC50 = 1090 nM T15556 CD5RM7 9962028 IC50 = 100 nM T15556 CN60FW 9970082 IC50 = 13000 nM T15556 C6TYV2 10076852 IC50 = 500 nM T15556 CY24DT 10099868 IC50 = 520 nM T15556 CBA32D 10108853 IC50 = 26000 nM T15556 CAL18T 10117515 IC50 > 50000 nM T15556 CQG17K 10138077 IC50 = 9800 nM T15556 C8LI2M 10160378 IC50 = 10000 nM T15556 CE7K1O 10163714 IC50 = 16000 nM T15556 CU6HX9 10203555 IC50 > 50000 nM T15556 CAQN51 10225186 IC50 = 17000 nM T15556 CT9K3A 10258248 IC50 = 390 nM T15556 CKG2M3 10297078 IC50 = 21000 nM T15556 CGD6J5 10410195 IC50 = 300 nM T15556 C7OI3J 10455506 IC50 = 600 nM T15556 C3POD1 10484357 IC50 = 530 nM T15556 C02GKL 11180570 IC50 = 8300 nM T15556 C13GPO 11192092 IC50 = 12000 nM T15556 CH5GZ7 11203757 IC50 = 23000 nM T15556 COX56M 11261201 IC50 = 28700 nM T15556 CQ9DE5 11261480 IC50 = 28000 nM T15556 CJS9C0 11304851 IC50 = 7900 nM T15556 C30YOT 11728770 IC50 = 700000 nM T15556 CAS68J 12019961 IC50 = 1930 nM T15556 CY59MK 15482075 IC50 = 10800 nM T15556 C1IQ5A 16770662 IC50 = 5200 nM T15556 CO0QH5 18364391 IC50 = 2910 nM T15556 CRJ1H4 18364393 IC50 = 240 nM T15556 CX7ZA5 18364403 IC50 = 2070 nM T15556 CIZQ03 18364405 IC50 = 39 nM T15556 CIP0A6 18364410 IC50 = 100 nM T15556 COK1S9 18364413 IC50 = 270 nM T15556 CL20PQ 24829269 IC50 = 5000 nM T15556 C25HDG 24829409 IC50 = 4500 nM T15556 CH23JG 24873595 IC50 = 14400 nM T15556 CY98BD 24873596 IC50 > 80000 nM T15556 CT0HC4 24873597 IC50 = 15400 nM T15556 CFVC76 24873598 IC50 = 25000 nM T15556 C4Z3BC 24873654 IC50 = 14900 nM T15556 CFGP62 24873655 IC50 = 8500 nM T15556 CR9LD4 24873656 IC50 = 61000 nM T15556 C3N4QI 24873730 IC50 = 8400 nM T15556 C48CTM 24873732 IC50 = 23000 nM T15556 CC2SU0 24873733 IC50 = 75000 nM T15556 C3SZ0U 24873734 IC50 = 29900 nM T15556 C29XNU 24873796 IC50 = 11000 nM T15556 CH94VA 24873797 IC50 = 9300 nM T15556 C9CR1S 24873798 IC50 = 114000 nM T15556 CV6MA4 24873799 IC50 = 21000 nM T15556 CVL80Q 24873860 IC50 = 43000 nM T15556 CJ9FI6 24873861 IC50 = 86000 nM T15556 CHPE31 24873862 IC50 = 5400 nM T15556 CMFD48 24873863 IC50 = 12800 nM T15556 CH2XY9 24873918 IC50 = 13300 nM T15556 C62PJS 25114330 IC50 = 518000 nM T15556 C5G3WD 25114332 IC50 = 9320 nM T15556 C1Y0BZ 25174437 IC50 = 7940 nM T15556 CY5ZN6 44235156 IC50 = 9600 nM T15556 C5RNT3 44250422 IC50 = 3550 nM T15556 C7LO2F 44250489 IC50 = 7450 nM T15556 C7R2HY 44251374 IC50 = 3560 nM T15556 CZM14A 44266596 IC50 = 200 nM T15556 CX8A1J 44292071 IC50 = 770 nM T15556 CIL50Y 44292073 IC50 = 470 nM T15556 C49EIC 44315428 IC50 = 12000 nM T15556 CU1N4I 44315429 IC50 = 4000 nM T15556 C85NED 44315448 IC50 = 23600 nM T15556 CZNL62 44315493 IC50 = 8600 nM T15556 CE4M6H 44315506 IC50 > 50000 nM T15556 CD52XE 44315507 IC50 = 18000 nM T15556 C2E1SJ 44315654 IC50 = 1000 nM T15556 CW0S4Q 44315704 IC50 = 9800 nM T15556 CV3Z9E 44315705 IC50 = 39500 nM T15556 C1GR7E 44315721 IC50 = 1900 nM T15556 CK0M4Q 44320713 IC50 = 1750 nM T15556 C6XF1H 44320731 IC50 = 20000 nM T15556 C3UQS5 44320742 IC50 > 25000 nM T15556 C1N3IF 44320743 IC50 > 25000 nM T15556 CQ24JL 44320756 IC50 = 15000 nM T15556 CT9F4E 44321072 IC50 = 12400 nM T15556 CS01QV 44321079 IC50 = 17700 nM T15556 C3D9YL 44321088 IC50 = 4770 nM T15556 C1BFR7 44321113 IC50 = 13100 nM T15556 CEH1L6 44321114 IC50 > 25000 nM T15556 CIN48S 44321153 IC50 = 10900 nM T15556 C1Y5OH 44321174 IC50 = 6100 nM T15556 CS69YB 44321183 IC50 > 25000 nM T15556 C5PBJ1 44321186 IC50 > 25000 nM T15556 CA1H9Z 44321192 IC50 = 3100 nM T15556 C3UE0M 44321195 IC50 > 25000 nM T15556 C9YEQ4 44321203 IC50 > 25000 nM T15556 CNZC21 44321205 IC50 > 25000 nM T15556 CW2DZ8 44321225 IC50 > 25000 nM T15556 CW9K0G 44341217 IC50 > 15000 nM T15556 CWC43M 44341277 IC50 = 2900 nM T15556 CD4BH6 44341290 IC50 = 890 nM T15556 C63QVZ 44341310 IC50 = 900 nM T15556 C6A2KF 44341356 IC50 = 3900 nM T15556 C7RIS6 44341370 IC50 = 1400 nM T15556 C2KBV3 44341400 IC50 = 1100 nM T15556 CC4XT2 44341438 IC50 = 1800 nM T15556 CMFJ89 44341459 IC50 = 2600 nM T15556 CA96RU 44341473 IC50 = 2900 nM T15556 C3GQ4W 44341477 IC50 = 2600 nM T15556 C9K6HM 44341493 IC50 = 100 nM T15556 CX1Z2N 44341495 IC50 = 2200 nM T15556 C0JT1G 44341503 IC50 > 15000 nM T15556 C85SYZ 44341504 IC50 > 15000 nM T15556 CC7U5X 44341509 IC50 = 940 nM T15556 CEO8H7 44341510 IC50 = 2700 nM T15556 CAN5E0 44341523 IC50 = 3200 nM T15556 CB98LY 44341603 IC50 = 600 nM T15556 COXM08 44341604 IC50 > 15000 nM T15556 CX51BU 44341605 IC50 = 5000 nM T15556 C3HU6I 44341630 IC50 = 1400 nM T15556 CWP6Q7 44341689 IC50 = 710 nM T15556 C26VDF 44341690 IC50 = 700 nM T15556 C9SGU5 44341691 IC50 = 710 nM T15556 CR1G8I 44341692 IC50 = 1400 nM T15556 CO4M6D 44341839 IC50 = 100 nM T15556 CFO69B 44341840 IC50 = 7800 nM T15556 C3JCN8 44341851 IC50 > 15000 nM T15556 C9Q6HW 44344073 IC50 = 10000 nM T15556 CBN2W3 44344205 IC50 = 35000 nM T15556 C4FP8D 44377761 IC50 = 3500 nM T15556 CYJ57W 44377766 IC50 = 900 nM T15556 CZEU62 44377767 IC50 = 1000 nM T15556 CUFW40 44377796 IC50 = 4300 nM T15556 C7FM5B 44377813 IC50 = 5000 nM T15556 C2PT7O 44377833 IC50 = 2800 nM T15556 C3TL6Q 44377858 IC50 > 15000 nM T15556 CE61RW 44377874 IC50 > 15000 nM T15556 CV3R1O 44377889 IC50 = 1800 nM T15556 CD3K0T 44378046 IC50 = 1500 nM T15556 CIG8X6 44378047 IC50 = 800 nM T15556 CLG5Q4 44378049 IC50 = 2100 nM T15556 C1C3EZ 44378050 IC50 = 900 nM T15556 C0RMV9 44378055 IC50 = 3400 nM T15556 C8N7BY 44378061 IC50 = 3200 nM T15556 CSC81G 44378063 IC50 = 1100 nM T15556 C56NTK 44378073 IC50 = 2800 nM T15556 CRQE86 44378075 IC50 = 880 nM T15556 CR1M5K 44378082 IC50 = 7900 nM T15556 CGS16U 44378083 IC50 = 500 nM T15556 C25FUD 44378084 IC50 = 1700 nM T15556 C3K4VQ 44378087 IC50 = 910 nM T15556 CNX1L0 44378181 IC50 > 15000 nM T15556 CMU7T1 44378197 IC50 = 3700 nM T15556 CDKU64 44378198 IC50 = 900 nM T15556 CKG8X5 44378200 IC50 = 1700 nM T15556 CO4G8M 44378232 IC50 = 6100 nM T15556 CI61QC 44378237 IC50 = 6700 nM T15556 C31NPK 44378270 IC50 = 1400 nM T15556 C3FYR7 44378271 IC50 = 700 nM T15556 CR3QB8 44378272 IC50 = 1700 nM T15556 CJW51U 44378273 IC50 = 1000 nM T15556 CP7O9Q 44397007 IC50 = 63100 nM T15556 C65AWE 44558994 IC50 = 138000 nM T15556 C7RD3H 44558995 IC50 = 152000 nM T15556 C3LMO2 44560368 IC50 = 96000 nM T15556 CY8FB5 46191021 IC50 = 650 nM T15556 C5Y1SR 46191086 IC50 = 690 nM T15556 C03IMY 46216724 IC50 = 284 nM T15556 CZB9H4 46216725 IC50 = 594 nM T15556 CKH1U4 46227800 IC50 = 1100 nM T15556 C04LSW 46227802 IC50 = 940 nM T15556 CKCH03 46227821 IC50 = 1200 nM T15556 C12QIT 46227824 IC50 = 1500 nM T15556 CV5HR2 46227825 IC50 = 7800 nM T15556 CEO59P 46231363 IC50 > 300000 nM T15556 C0R7FE 46231364 IC50 > 300000 nM T15556 CI2Q9S 46231365 IC50 > 300000 nM T15556 C3Y0ZF 46231366 IC50 = 128000 nM T15556 CTJ7M6 46231367 IC50 = 2670 nM T15556 CQL8T5 46231408 IC50 = 4820 nM T15556 CNGE41 46232215 IC50 > 300000 nM T15556 CW83FO 46232293 IC50 > 3000000 nM T15556 C9OM5J 46232294 IC50 = 1384000 nM T15556 CG5P2S 46232295 IC50 > 300000 nM T15556 CYCT81 46232296 IC50 = 343000 nM T15556 C8KL6M 46935552 IC50 = 2820 nM T15556 CQ2C1M 46935554 IC50 = 7390 nM T15556 C93FMN 46935597 IC50 = 2420 nM T15556 CUO05N 53483962 IC50 = 3200 nM T15556 C4WH7T 54680250 IC50 = 1650 nM T15556 C6PS7F 54682797 IC50 = 4250 nM T15556 C8RGO6 54715796 IC50 = 510 nM T15556 CW7T4A 54720084 IC50 = 2200 nM T15556 C7IAC3 54730495 IC50 = 24000 nM T15556 CN30IK 54730496 IC50 = 13700 nM T15556 CE3G1R 54730497 IC50 = 1000 nM T15556 C9K8ED 54730498 IC50 = 14000 nM T15556 C2UXN7 54731757 IC50 = 300 nM T15556 C78EHL 54731758 IC50 = 900 nM T15556 CJQS07 54731760 IC50 = 1950 nM T15556 CW90BM 54731762 IC50 > 50000 nM T15556 C4H1TR 54731763 IC50 = 7000 nM T15556 CC0OR3 54731764 IC50 = 1850 nM T15556 C5U9WB 54731765 IC50 = 3000 nM T15556 C3I9FM 54731767 IC50 = 1030 nM T15556 CZ8F9R 54731769 IC50 = 600 nM T15556 CAQT09 54731770 IC50 = 670 nM T15556 CX09NI 54731771 IC50 = 2000 nM T15556 C9R2EV 54731773 IC50 = 7900 nM T15556 C8LPC4 54731775 IC50 > 30000 nM T15556 C6WO1Q 54731777 IC50 = 4900 nM T15556 CC68DB 54731779 IC50 = 1010 nM T15556 CLH43E 54731780 IC50 = 30000 nM T15556 CO3B5G 54731781 IC50 > 20000 nM T15556 CX86KA 54731782 IC50 = 3600 nM T15556 C5SO3T 54731783 IC50 = 1800 nM T15556 CO82IC 54735311 IC50 = 500 nM T15556 CKX65J 54735313 IC50 = 2350 nM T15556 CA3D2E 56658166 IC50 = 98000 nM T15556 CXZC82 56658167 IC50 = 29000 nM T15556 C3IRZ7 56658168 IC50 = 2400 nM T15556 C49ORE 56661678 IC50 = 4900 nM T15556 C8Q2CU 56665087 IC50 = 3400 nM T15556 C49TWH 56665088 IC50 = 14600 nM T15556 C8I2EZ 56672040 IC50 = 22000 nM T15556 C43KNI 56682076 IC50 = 63800 nM T15556 CC1DN7 60008645 IC50 = 4110 nM T15556 C73VIT 66679603 IC50 > 20000 nM T15556 C0N7WB 66679802 IC50 > 40000 nM T15556 CY43MI 66680045 IC50 = 1860 nM T15556 CFJ3W2 66680174 IC50 = 3190 nM T15556 C3HO7I 66680327 IC50 = 4740 nM T15556 CT20IU 66680337 IC50 = 900 nM T15556 COKQ96 66680370 IC50 = 5520 nM T15556 C0YOT4 66680377 IC50 = 7800 nM T15556 C1TRL0 66680380 IC50 = 2310 nM T15556 C3AGJ1 66680426 IC50 = 2400 nM T15556 CM7W3E 66680617 IC50 = 1170 nM T15556 CY53HN 66680639 IC50 = 1670 nM T15556 C86SHF 66680788 IC50 = 3630 nM T15556 C0KW3Y 66680861 IC50 = 2980 nM T15556 CW19QL 66680871 IC50 = 1840 nM T15556 CJA78X 66681185 IC50 = 6410 nM T15556 C1DR8M 145965481 IC50 > 10000 nM T15556 C9W8UZ 145976402 IC50 = 21600 nM T15556 D05GSZ 10479348 IC50 = 13000 nM T15556 D05VKW 10413640 IC50 = 4700 nM T15556 D0U4LV 9848832 IC50 = 5300 nM T15556 D0WX7S 10391273 IC50 = 3300 nM T29754 D0EG1I 9926791 IC50 > 10000 nM T29754 D03LWG 53235510 IC50 > 10000 nM T29754 D07EHV 44814409 IC50 > 10000 nM T29754 D07HPJ 11476171 IC50 > 10000 nM T29754 D0E3TC 44259 IC50 = 295 nM T29754 D0U2BH 65064 IC50 = 1000 nM T29754 D03BNU 59604787 IC50 > 10000 nM T29754 D0R1JI 5281847 IC50 = 1900 nM T29754 D0T3ME 156422 IC50 > 30000 nM T29754 CJWX69 3848929 IC50 = 19000 nM T29754 CL5I2U 5330279 IC50 > 10000 nM T29754 CM5Z8X 9869943 IC50 > 1000 nM T29754 C2Y3WG 9907612 IC50 = 11000 nM T29754 CJO47T 9948405 IC50 > 10000 nM T29754 CV8I5X 9999342 IC50 > 10000 nM T29754 C5TQ7X 10247543 IC50 > 10000 nM T29754 C2WQ8M 10473563 IC50 > 10000 nM T29754 C0APW4 11422034 IC50 > 10000 nM T29754 CU0E8O 11690457 Ki > 10000 nM T29754 CB0AP2 11705863 Ki > 10000 nM T29754 C8E4TS 11992146 IC50 = 210 nM T29754 C9TU1O 16046126 IC50 > 1000 nM T29754 CUR7H3 16719862 IC50 = 140 nM T29754 CG6D4M 23647319 IC50 > 10000 nM T29754 CY8Z7X 23647330 IC50 > 10000 nM T29754 C4XD8H 23647348 IC50 > 10000 nM T29754 CDMI50 23661564 IC50 = 24000 nM T29754 C7YG1N 24759534 IC50 = 9600 nM T29754 CLBP72 24798571 IC50 > 10000 nM T29754 CQ3Y4R 24856513 IC50 = 914 nM T29754 CA5D6Q 24856601 IC50 > 10000 nM T29754 CPC3V6 24856688 IC50 > 10000 nM T29754 C2W8HA 24857177 IC50 = 1490 nM T29754 CKV0D5 24857447 IC50 = 390 nM T29754 CWX59J 24857738 IC50 = 829 nM T29754 CY8L7E 24896769 IC50 > 10000 nM T29754 C9URB7 44441149 IC50 = 25000 nM T29754 C4IY8M 45256689 IC50 < 10000 nM T29754 CLS29B 46872626 IC50 > 10000 nM T29754 C2B5XF 49765254 IC50 > 10000 nM T29754 CJZ5A0 49840306 IC50 > 10000 nM T29754 CRA74I 49842779 IC50 > 10000 nM T29754 CEQN27 52936621 Ki > 1000 nM T29754 C8NA4L 53384644 IC50 > 30000 nM T29754 C1XS2J 54760383 IC50 > 10000 nM T29754 C0LSM5 57345529 IC50 = 195 nM T29754 C9X3UG 57390456 IC50 = 2390 nM T29754 C9EH0V 57392242 IC50 > 10000 nM T29754 C8AE5I 57393992 IC50 = 3200 nM T29754 CG2H9V 57393993 IC50 = 239 nM T29754 CM5B4Z 57394002 IC50 = 290 nM T29754 C1AEY9 57395762 IC50 = 3730 nM T29754 CEF15U 57395763 IC50 = 88 nM T29754 CP27IV 57397535 IC50 > 10000 nM T29754 CSUN39 57399215 IC50 > 10000 nM T29754 C6XN4M 57399216 IC50 = 437 nM T29754 CR7PC5 57400976 IC50 = 392 nM T29754 CV3J8L 57400977 IC50 = 2820 nM T29754 CB3CT5 57402741 IC50 = 148 nM T29754 CXJ63M 59603829 IC50 = 19000 nM T29754 CQEU96 59603842 IC50 = 1400 nM T29754 C1HSE0 67035086 IC50 = 3700 nM T29754 CWI6K5 67035106 IC50 > 10000 nM T29754 C38RGB 67035556 IC50 > 10000 nM T29754 CV63UL 67240318 IC50 > 10000 nM T29754 C8I7GC 68293638 IC50 > 10000 nM T29754 C5DGR9 69036886 IC50 = 10000 nM T29754 C1IEJ2 70789254 IC50 = 226000 nM T29754 C8T7ZP 70789255 IC50 = 41000 nM T29754 CJ2T9E 76332983 IC50 > 10000 nM T29754 C1HW4B 89735655 IC50 > 100000 nM T29754 CTJ48K 135524085 IC50 = 28 nM T29754 CUT1W7 135524168 IC50 = 24 nM T29754 C27RQE 135979614 IC50 = 816 nM T29754 C6VB3O 145925651 IC50 >= 5000 nM T29754 D00ERW 44444843 Ki > 1525 nM T29754 D03DZO 11715767 IC50 = 500 nM T29754 D06HVH 54613583 IC50 = 1700 nM T29754 D0EW9J 10389239 IC50 = 81 nM T29754 D0GD8Y 3006531 IC50 = 50000 nM T85733 D03NHW 4583 IC50 = 1 ug.mL-1 T85733 D07JGT 4421 IC50 = 52 ug.mL-1 T85733 D07VLY 31703 IC50 = 3500 nM T85733 D0B7EB 36462 IC50 = 69.8 nM T85733 D0G9YH 2179 IC50 = 2760 nM T85733 D0O1WX 2764 IC50 = 0.3 ug.mL-1 T85733 D0Q2PE 4539 IC50 = 1 ug.mL-1 T85733 D0PM9P 6918093 IC50 = 0.31 ug.mL-1 T85733 CO25YL 62999 IC50 = 0.2 ug.mL-1 T85733 CY16ER 130078 EC50 > 54000 nM T85733 CH34KQ 194999 IC50 = 1 ug.mL-1 T85733 C2P6EC 372648 EC50 > 50000 nM T85733 C13OPQ 5352088 IC50 = 101200 nM T85733 CL9BG2 9910942 EC50 = 930 nM T85733 C4DB6I 9956691 IC50 = 58.3 ug.mL-1 T85733 CMAO97 10367045 IC50 = 95 ug.mL-1 T85733 C4EM6S 10426517 EC50 > 55000 nM T85733 CE8D4G 10433396 IC50 = 0.4 ug.mL-1 T85733 CULK80 10555744 IC50 = 0.2 ug.mL-1 T85733 CMLX35 10556110 IC50 = 40 ug.mL-1 T85733 CR1L5K 10594738 IC50 > 500 ug.mL-1 T85733 C7Q0MZ 10694889 IC50 > 500 ug.mL-1 T85733 CR3CO8 10697323 IC50 > 500 ug.mL-1 T85733 CB38HW 10719596 IC50 = 658 ug.mL-1 T85733 CM27IA 11089787 IC50 = 25.6 ug.mL-1 T85733 CCG3Y1 11456414 IC50 = 0.1 ug.mL-1 T85733 CVK85X 11725233 IC50 = 0.59 ug.mL-1 T85733 CRY8D3 13652996 IC50 = 0.16 ug.mL-1 T85733 CQ8YG0 13652997 IC50 = 1.2 ug.mL-1 T85733 CA8I1R 14390997 IC50 = 0.17 ug.mL-1 T85733 CSN9C7 14390999 IC50 = 0.31 ug.mL-1 T85733 CCX8O3 14391001 IC50 = 0.93 ug.mL-1 T85733 CHF78C 14391002 IC50 = 0.35 ug.mL-1 T85733 CPL38S 14391003 IC50 = 0.25 ug.mL-1 T85733 CI0E2S 18654132 EC50 > 50000 nM T85733 C2GZ7E 44352936 EC50 > 60000 nM T85733 CL97SM 44353499 EC50 > 50000 nM T85733 CVWY40 44353548 EC50 > 51000 nM T85733 CWDO54 44353588 EC50 > 50000 nM T85733 CA20OD 44353638 EC50 > 60000 nM T85733 C0HXQ4 44353647 EC50 > 50000 nM T85733 CH78SF 44353648 EC50 > 50000 nM T85733 C8QPD4 44353654 EC50 > 50000 nM T85733 CUYJ90 44353655 EC50 > 60000 nM T85733 CPEW14 44353667 EC50 = 1200 nM T85733 C0Q1CK 44353715 EC50 = 27000 nM T85733 CXQ5D4 44353853 EC50 > 60000 nM T85733 CC90EW 44353863 EC50 > 60000 nM T85733 C7CPN8 44355399 IC50 = 12500 nM T85733 CL3YD1 54729892 IC50 = 10.3 ug.mL-1 T85733 CH2MB6 54731796 IC50 = 49 ug.mL-1 T85733 C2LXW4 54731797 IC50 = 30 ug.mL-1 T85733 CVT4U2 54731802 IC50 = 100 ug.mL-1 T85733 CU43YS 54731809 IC50 = 3.5 ug.mL-1 T85733 CEQV69 54731812 IC50 = 64 ug.mL-1 T85733 CDS29Y 54731813 IC50 = 17 ug.mL-1 T85733 C0ACN9 54731814 IC50 = 31 ug.mL-1 T85733 CM9GI6 145949253 IC50 = 81.42 nM T85733 C12UAN 145951484 IC50 = 12.6 nM T85733 C5GZ9J 145954861 IC50 = 110.45 nM T85733 CL01ST 145959691 IC50 = 6.85 nM T85733 C4SK8I 145962714 IC50 = 31.68 nM T85733 C73KTM 145966514 IC50 = 580 nM T85733 C7EO5Q 145976349 IC50 = 860 nM T85733 CAK6O4 145981649 IC50 = 9290 nM T85733 C2JRE3 155519532 IC50 = 4340 nM T85733 CL2KQ5 155532817 IC50 = 5250 nM T85733 CTW37I 155555640 IC50 = 1060 nM T85733 C83GLS 155563816 IC50 = 1150 nM T85733 D00DXV 9895647 IC50 = 0.4 ug.mL-1 T85733 D03NXV 2134 IC50 = 30 nM T35809 CZ3Y9X 2972356 IC50 = 2050 nM T35809 C42AQR 4102773 IC50 = 450 nM T35809 CTU52G 49190366 IC50 = 6140 nM T35809 CM6Y4O 49190451 IC50 = 4300 nM T35809 CIS4D7 49190466 IC50 = 1710 nM T35809 CDQ80N 50796602 IC50 = 2770 nM T35809 CYP58I 50796734 IC50 = 3470 nM T35809 CX12UC 50796762 IC50 = 1210 nM T35809 C2GP8Q 50796763 IC50 = 5160 nM T35809 C5UQ8O 50796790 IC50 = 1330 nM T35809 CP1U8X 50796792 IC50 = 2380 nM T35809 C1R7BG 50796818 IC50 > 10000 nM T35809 CT34KZ 50796842 IC50 = 2390 nM T35809 CTSH48 50796873 IC50 = 2420 nM T35809 CA01UQ 50796897 IC50 = 3690 nM T35809 CPZ93K 50820616 IC50 > 10000 nM T35809 CA2MT4 50820637 IC50 = 3580 nM T35809 CVG1Y0 50820716 IC50 = 2920 nM T35809 CG3PR6 52912222 IC50 > 19952.62 nM T35809 C76ZPW 71271926 IC50 = 130 nM T35809 CIPN50 71760902 IC50 > 1000 nM T35809 C5TB9S 77843982 IC50 > 1000 nM T35809 COME25 118918694 IC50 = 6700 nM T35809 CF9J8E 118918705 IC50 = 80 nM T35809 CA3Z8O 118918714 IC50 = 200 nM T35809 C8GLJ3 118918720 IC50 = 450 nM T35809 CAZR96 118918740 IC50 = 510 nM T35809 C37ZJX 118932971 IC50 = 230 nM T35809 C4DF6I 118932972 IC50 = 270 nM T35809 C2ZY3U 118932975 IC50 = 520 nM T35809 C2O0NE 118932978 IC50 = 1700 nM T35809 CHCU32 118932979 IC50 = 380 nM T35809 C2JCY3 118932989 IC50 = 150 nM T35809 CC14FI 118933132 IC50 = 48 nM T35809 CEPT12 118933133 IC50 = 100 nM T35809 CKY8H3 118933134 IC50 = 190 nM T35809 CGO91Y 118933136 IC50 = 1800 nM T35809 CC35IE 118933137 IC50 = 150 nM T35809 CBD7I6 121232405 IC50 = 7943.28 nM T35809 CM8UD0 121232406 IC50 = 50118.72 nM T35809 CWJD15 122705990 IC50 = 6 nM T35809 CM8EB4 126961333 IC50 = 94 nM T35809 CZ8S4U 127025422 IC50 = 2460 nM T35809 CB3RH7 127025423 IC50 > 10000 nM T35809 C6TY8H 127025698 IC50 = 1600 nM T35809 CTX9Y6 127029368 IC50 = 1700 nM T35809 CT93VU 127029369 IC50 = 1990 nM T35809 CFH9G7 127029370 IC50 = 2670 nM T35809 C7NEB1 130471695 IC50 = 1500 nM T35809 CLA09E 130471696 IC50 = 124 nM T35809 CWNY27 130471723 IC50 = 66 nM T35809 CXW1B4 130471724 IC50 = 1240 nM T35809 C1EN7A 130471730 IC50 = 121 nM T35809 C2HD6P 130471733 IC50 = 95 nM T35809 C5DFI7 130471761 IC50 = 366 nM T35809 CDLE96 130471765 IC50 = 153 nM T35809 C1C8OB 130471770 IC50 = 51 nM T35809 CDC32I 130471775 IC50 = 102 nM T35809 C3D7HE 130471777 IC50 = 248 nM T35809 CFI30C 130471784 IC50 = 84 nM T35809 C7TJA6 130471785 IC50 = 61 nM T35809 CDUX50 130471789 IC50 = 80 nM T35809 C8VAM6 130471790 IC50 = 74 nM T35809 CN80UV 130471849 IC50 = 82 nM T35809 CEV5I3 130471855 IC50 = 675 nM T35809 CE1K3M 130471876 IC50 = 70 nM T35809 CFTG42 130472058 IC50 = 63 nM T35809 C5P2ED 130472268 IC50 = 915 nM T35809 C7B6CZ 130472269 IC50 = 126 nM T35809 CED70X 130472274 IC50 > 10000 nM T35809 CK0B6N 131985884 IC50 = 1400 nM T35809 CPWF20 137632687 IC50 = 4400 nM T35809 CD4NE1 137633137 IC50 = 3300 nM T35809 CQT3A9 137636309 IC50 > 100000 nM T35809 CCAP49 137636933 IC50 = 100 nM T35809 CV1EP8 137639742 IC50 = 7800 nM T35809 CC3VL8 137644086 IC50 = 14000 nM T35809 CC34KQ 137650533 IC50 = 2600 nM T35809 CQ6XB7 139030526 IC50 = 12589.25 nM T35809 D03BTJ 15990224 IC50 = 7943.28 nM T35809 D08RDI 35397514 IC50 = 1200 nM T35809 D0C2PD 50796983 IC50 = 1750 nM T35809 D0O6XT 91827373 IC50 = 619 nM T35809 D0Q7IU 40642506 IC50 = 1110 nM T51115 D00STL 644241 IC50 = 199526.23 nM T51115 D01AXB 60835 IC50 = 25118.86 nM T51115 D01AZG 5073 IC50 = 125000 nM T51115 D03FLC 3878 IC50 = 1258925.41 nM T51115 D03IGH 213039 IC50 = 1584893.19 nM T51115 D03QWT 73303 IC50 = 1995.26 nM T51115 D04FVU 6337614 IC50 = 398107.17 nM T51115 D04JEE 4946 IC50 = 21000 nM T51115 D04OSE 4485 Ki = 1 nM T51115 D04VMT 5253 IC50 = 1023000 nM T51115 D05MQK 110635 IC50 = 398107.17 nM T51115 D05OFX 219078 IC50 = 50118.72 nM T51115 D06XMU 6013 IC50 = 34 nM T51115 D08CDI 208908 IC50 = 1995262.31 nM T51115 D08JIV 2162 IC50 = 1200 nM T51115 D08QMX 5757 IC50 = 50000 nM T51115 D09GOS 2812 IC50 = 590 nM T51115 D09MWJ 2092 IC50 = 199526.23 nM T51115 D0B3UJ 115237 IC50 = 398107.17 nM T51115 D0BZ7W 443879 IC50 = 25118.86 nM T51115 D0C9SY 135400189 IC50 = 15848.93 nM T51115 D0D7KC 5488548 IC50 = 5011.87 nM T51115 D0D8VE 3562 IC50 = 1800000 nM T51115 D0E4DW 1775 IC50 = 125000 nM T51115 D0E6XR 3062316 IC50 = 251188.64 nM T51115 D0L4YD 154059 IC50 = 6309.57 nM T51115 D0NW3X 71329 IC50 = 158489.32 nM T51115 D0OB1J 39186 IC50 = 44000 nM T51115 D0Q5UQ 214348 IC50 = 1000000 nM T51115 D0R0FE 2520 IC50 = 23500 nM T51115 D0R0MW 5329102 IC50 = 199526.23 nM T51115 D0S5CU 4499 IC50 = 3 nM T51115 D0T0KA 4474 IC50 = 250 nM T51115 D0U0VU 5312125 IC50 = 794328.23 nM T51115 D0U1OE 5452 IC50 = 1320 nM T51115 D0U2JP 4369359 IC50 = 100000000 nM T51115 D0X5ZI 6918493 IC50 = 2511886.43 nM T51115 D0Y4JJ 2351 IC50 = 1400 nM T51115 D0Y5AM 444031 IC50 = 1584893.19 nM T51115 D0Z1UA 71301 IC50 = 15848.93 nM T51115 D0Z7KE 3784 IC50 = 2.2 nM T51115 D0Z7ZM 135398744 IC50 = 100000 nM T51115 D00ERV 1234 IC50 = 17 nM T51115 D05ADP 160355 IC50 = 23400 nM T51115 D06ENM 66553195 IC50 = 36000 nM T51115 D0DH5X 44472635 IC50 > 30000 nM T51115 D0I2XM 3038500 IC50 = 1700 nM T51115 D0L9QM 59568713 IC50 > 30000 nM T51115 D0M3XR 46209133 IC50 > 30000 nM T51115 D0N3SR 5282138 IC50 = 5300 nM T51115 D0S5IR 86294073 IC50 > 30000 nM T51115 D0W8XT 60663 IC50 = 202 nM T51115 D08SOF 5405 IC50 = 1320 nM T51115 CTI3W4 40704 IC50 = 1750 nM T51115 CB31NV 60065 IC50 = 4900 nM T51115 CT15HN 341862 Ki = 27.1 nM T51115 CURH47 341863 Ki = 13.9 nM T51115 CLD6J9 441074 IC50 = 19820 nM T51115 CGY61C 443869 IC50 = 1200 nM T51115 CZN6S9 743974 IC50 > 15848.93 nM T51115 C1AQ4G 2870439 IC50 > 10000 nM T51115 C8KN4J 3876755 IC50 > 10000 nM T51115 CZ8TQ5 3944785 IC50 > 10000 nM T51115 CW2UD8 4099361 IC50 = 3200 nM T51115 CJO8N6 10117450 IC50 = 347 nM T51115 CSRI97 10413420 IC50 = 260 nM T51115 CK6N9E 13181322 Ki = 28.5 nM T51115 C1I8XD 13567332 Ki = 30 nM T51115 C0S6IR 13567333 Ki = 650 nM T51115 CYQ91M 13567337 Ki = 6000 nM T51115 CG9F8Y 13567338 Ki = 250 nM T51115 CQO2A3 13755646 Ki = 1 nM T51115 CK8Z7C 13755648 Ki = 80 nM T51115 C1X4MY 13763172 Ki = 505 nM T51115 CD34SB 15982534 IC50 = 92000 nM T51115 CG8KR9 16005860 IC50 = 14900 nM T51115 CE7DV0 23661730 IC50 = 3500 nM T51115 CX8DH1 24769723 IC50 > 30000 nM T51115 C91QFN 25019282 IC50 > 30000 nM T51115 C1IW5M 25261456 IC50 > 10000 nM T51115 CX4YL8 44232522 IC50 > 30000 nM T51115 C7UY5F 44235863 IC50 > 30000 nM T51115 CX2W8Y 44236320 IC50 = 15000 nM T51115 C8LN0U 44236321 IC50 = 30000 nM T51115 CK4S5Y 44236322 IC50 > 30000 nM T51115 CJX27R 44318678 IC50 = 250 nM T51115 CHA52K 44318895 IC50 = 270 nM T51115 C9Z1ST 44318909 IC50 = 100 nM T51115 CU85CR 44359060 IC50 = 410 nM T51115 CE9DS0 44442675 IC50 = 1725 nM T51115 C2QK4J 44472590 IC50 = 8200 nM T51115 CQ8C3F 44472591 IC50 = 13000 nM T51115 CC2TA5 44472592 IC50 > 30000 nM T51115 CWN95E 44472610 IC50 > 30000 nM T51115 C1H2ZT 44472612 IC50 > 30000 nM T51115 C9G5ID 44472613 IC50 > 30000 nM T51115 C5N4KE 44472633 IC50 > 30000 nM T51115 C1FTA7 44481065 IC50 > 30000 nM T51115 C6HTC1 44583235 IC50 > 30000 nM T51115 C5SI9Q 44583288 IC50 > 30000 nM T51115 CC19TZ 44583290 IC50 = 20000 nM T51115 C90RAV 44583349 IC50 = 28000 nM T51115 CK81NJ 44583350 IC50 = 26000 nM T51115 CUT2B4 45267348 IC50 > 30000 nM T51115 CJH3A2 45268206 IC50 > 30000 nM T51115 C4WR0V 45269087 IC50 > 30000 nM T51115 CRPS25 45269096 IC50 > 30000 nM T51115 C7BNY6 45269104 IC50 = 2000 nM T51115 CS1Q2X 45269947 IC50 > 30000 nM T51115 C1BE5U 45269948 IC50 > 30000 nM T51115 CG1H9N 45269950 IC50 = 12000 nM T51115 C1NT2M 45270771 IC50 > 30000 nM T51115 CA05IG 45270778 IC50 > 30000 nM T51115 CZ7MK9 45270788 IC50 = 3000 nM T51115 C9TM2P 45271593 IC50 = 11000 nM T51115 C06YAD 45271599 IC50 > 30000 nM T51115 CG0I8P 45271610 IC50 > 30000 nM T51115 C6FBH0 45271618 IC50 = 6800 nM T51115 C71VIG 45272510 IC50 = 19000 nM T51115 C05EDY 45272511 IC50 > 30000 nM T51115 CD62AH 45273373 IC50 > 30000 nM T51115 CMN39U 45273380 IC50 > 30000 nM T51115 C1ATC9 46203893 IC50 = 437 nM T51115 CHTV13 46203894 IC50 = 455 nM T51115 CFYP54 46203897 IC50 = 387 nM T51115 C9L4KT 46205341 IC50 > 333000 nM T51115 CL41FE 46206000 IC50 > 333000 nM T51115 C0SNL2 46209134 IC50 > 30000 nM T51115 CU63QR 49847377 IC50 > 20000 nM T51115 CJ7H2B 49847753 IC50 > 10000 nM T51115 C05SEW 49849008 IC50 > 20000 nM T51115 C78SAD 49849115 IC50 > 10000 nM T51115 CT3F0N 53235532 IC50 = 20000 nM T51115 CQIY23 53248846 IC50 > 30000 nM T51115 C9MHR0 53248847 IC50 = 25600 nM T51115 CJ83EB 53311393 IC50 > 10000 nM T51115 CPS12B 53317097 IC50 > 30000 nM T51115 CG69CQ 53327817 IC50 > 30000 nM T51115 C28RDF 54746913 IC50 > 30000 nM T51115 C6PUX9 56645570 IC50 > 30000 nM T51115 C1IY0P 56944164 IC50 > 20000 nM T51115 C4E1NK 57331209 IC50 > 100000 nM T51115 C9S8MU 57386524 IC50 > 10000 nM T51115 C3N4MF 57520842 IC50 > 30000 nM T51115 CEL56T 57520942 IC50 > 30000 nM T51115 CCQM76 59153288 IC50 > 30000 nM T51115 C2LBW7 66551925 IC50 > 30000 nM T51115 CL1RV4 67447319 IC50 = 424 nM T51115 CJ7FG0 67448236 IC50 = 533 nM T51115 CC9S6H 67449145 IC50 = 2670 nM T51115 CJ06LD 70683064 Ki = 3000 nM T51115 C46RHS 70685148 Ki = 500 nM T51115 CMVH17 70691450 Ki = 5000 nM T51115 C9AXI7 70695682 Ki = 5000 nM T51115 CBDL19 70792359 IC50 > 30000 nM T51115 CLIH32 71226367 IC50 = 4500 nM T51115 C6BE5X 71271461 IC50 > 30000 nM T51115 CA07TC 71517197 IC50 > 31600 nM T51115 C9J0EH 71603917 IC50 > 30000 nM T51115 C30NBJ 71722055 IC50 > 30000 nM T51115 CW20HQ 71818431 IC50 = 10000 nM T51115 C2L7TX 71818575 IC50 = 10000 nM T51115 C29YGC 72712370 IC50 > 100000 nM T51115 C3TXQ5 76321521 IC50 = 5900 nM T51115 CR05PL 76322043 IC50 > 30000 nM T51115 CQ3CW1 76322044 IC50 > 30000 nM T51115 C2YIP6 76332364 IC50 = 5420 nM T51115 C92WBQ 76336500 IC50 > 30000 nM T51115 C34TAM 77845572 IC50 = 18000 nM T51115 C2NCH9 78318214 IC50 = 22000 nM T51115 C2GET7 78318815 IC50 > 30000 nM T51115 CP8X3E 89573118 IC50 > 10000 nM T51115 C47HED 89583208 IC50 > 10000 nM T51115 C2BM9L 89768534 IC50 = 5700 nM T51115 C26LKW 90341025 IC50 = 18000 nM T51115 CZ62GY 118560409 IC50 = 7100 nM T51115 CB41MH 118560618 IC50 = 2410 nM T51115 CS0RQ3 118560699 IC50 = 2420 nM T51115 COIY31 118738348 IC50 = 70 nM T51115 CU4CW1 121313969 IC50 > 30000 nM T51115 CO9SQ6 121454909 IC50 > 30000 nM T51115 CH0X4Z 121454982 IC50 = 15000 nM T51115 CT0KS4 121455652 IC50 = 19000 nM T51115 CW35TI 121455794 IC50 = 15000 nM T51115 CHD26A 121596332 IC50 > 33300 nM T51115 CNGQ19 122179477 IC50 > 30000 nM T51115 C7KNL3 122187207 IC50 = 403 nM T51115 CYE4O0 122187208 IC50 = 156 nM T51115 C8Y5VF 122187209 IC50 = 225 nM T51115 CJ5OR3 122187210 IC50 = 504 nM T51115 CR5TW0 122187211 IC50 = 426 nM T51115 CA89DJ 122187212 IC50 = 748 nM T51115 CR2Q6E 122187213 IC50 = 140 nM T51115 CA3K1Y 122187853 IC50 > 4600 nM T51115 CI1NX6 122187854 IC50 = 434 nM T51115 C91RFU 122187855 IC50 = 173 nM T51115 CN7I3U 122187856 IC50 = 588 nM T51115 C1XKA8 122191834 IC50 > 30000 nM T51115 CIQ23U 126740608 IC50 = 1100 nM T51115 C1O5VB 126740610 IC50 = 1480 nM T51115 C9KEY6 126740618 IC50 = 2080 nM T51115 COE64S 126740626 IC50 = 3310 nM T51115 C4D9QY 127026491 IC50 > 30000 nM T51115 CKSZ13 127035240 IC50 > 30000 nM T51115 C7L1DB 127037832 IC50 > 30000 nM T51115 CO1RW6 134132142 IC50 = 12840 nM T51115 CS0A8O 134132803 IC50 = 8600 nM T51115 C58IKL 134133106 IC50 > 10000 nM T51115 C40FOB 134133525 IC50 > 10000 nM T51115 CJOQ95 134134229 IC50 = 15090 nM T51115 CS6Z7U 134135105 IC50 = 5900 nM T51115 CC7OQ2 134135307 IC50 > 30000 nM T51115 CE5TV4 134135453 IC50 = 21000 nM T51115 CMQV20 134136121 IC50 > 10000 nM T51115 C4SB8F 134136300 IC50 = 3600 nM T51115 CK9MG1 134136380 IC50 = 6400 nM T51115 C5VG6N 134136586 IC50 > 10000 nM T51115 C3W6FX 134137496 IC50 > 10000 nM T51115 CW5T6X 134138179 IC50 = 1880 nM T51115 CSEW05 134139055 IC50 = 2200 nM T51115 CAFS70 134139103 IC50 > 10000 nM T51115 C07AWK 134139327 IC50 > 10000 nM T51115 CQ6V1Z 134140414 IC50 = 7800 nM T51115 C9IMS2 134140658 IC50 = 2360 nM T51115 CZ06DO 134141633 IC50 = 4800 nM T51115 C4KI8G 134142247 IC50 > 10000 nM T51115 CTIX18 134145629 IC50 > 10000 nM T51115 CT0KP6 134146400 IC50 = 1340 nM T51115 CHF36J 134147928 IC50 = 2650 nM T51115 C1WSQ6 134148112 IC50 = 1940 nM T51115 C36CTV 134149105 IC50 > 10000 nM T51115 CRBG97 134149384 IC50 > 10000 nM T51115 CM9ZY1 134150199 IC50 > 10000 nM T51115 CA5B2J 134150245 IC50 > 30000 nM T51115 CJQ37D 134150323 IC50 = 2180 nM T51115 CI58UE 134150489 IC50 = 5700 nM T51115 CW38EV 134150541 IC50 > 10000 nM T51115 COPA84 134151189 IC50 > 30000 nM T51115 CPB68S 134152614 IC50 = 5400 nM T51115 CI61JC 134153846 IC50 = 3900 nM T51115 CFX72G 134154056 IC50 = 6300 nM T51115 CUH82M 134155661 IC50 = 3090 nM T51115 CA49BH 134156727 IC50 = 28000 nM T51115 C3O9IA 134156846 IC50 > 10000 nM T51115 C3TW0A 134374895 IC50 > 10000 nM T51115 CY4MV6 135566354 IC50 > 30000 nM T51115 CRPQ42 136069494 IC50 > 10000 nM T51115 C4OVP2 136416802 IC50 > 30000 nM T51115 C7ZCT8 136416815 IC50 > 30000 nM T51115 C6B5US 137628648 IC50 > 10000 nM T51115 CTD69B 137647980 IC50 = 4500 nM T51115 COLY80 137649218 IC50 = 13000 nM T51115 C8BDX5 137655281 IC50 = 8000 nM T51115 CE79SV 138377584 IC50 > 15000 nM T51115 CSJV78 145965046 IC50 = 2800 nM T51115 C74GDJ 145965861 IC50 = 860 nM T51115 C8RFM3 145973261 IC50 > 33000 nM T51115 CGW6Q5 145978668 IC50 = 2730 nM T51115 CY8IF4 145981627 IC50 > 10000 nM T51115 CU0K2Y 145990810 IC50 > 10000 nM T51115 CG8I5F 155538033 IC50 > 33000 nM T51115 C5T9KE 155542416 IC50 > 30000 nM T51115 C8Q2FG 155555556 IC50 = 16230 nM T51115 C3WT2Q 155556441 IC50 > 30000 nM T51115 CC5FE7 155564581 IC50 > 30000 nM T51115 CUT84A 155568798 IC50 > 30000 nM T51115 D0R6MT 3758 IC50 = 466000 nM T66925 D03ZFG 5282054 IC50 = 4000 nM T66925 D0J4IP 11433028 IC50 = 105000 nM T66925 D0KK6L 11202494 IC50 = 620 nM T66925 D0UR1H 71459385 IC50 = 67000 nM T66925 CK80QG 195372 IC50 = 100 nM T66925 CZT8Q4 263609 IC50 = 2400 nM T66925 CEIB95 2836767 IC50 > 100000 nM T66925 CGD0T7 6736443 IC50 > 80000 nM T66925 C14ZDI 10127128 IC50 = 1900 nM T66925 CHSE82 10151123 IC50 = 910 nM T66925 CE8TY5 10172880 IC50 = 2200 nM T66925 C05DAT 10194682 IC50 = 130 nM T66925 CNH43O 10215862 IC50 = 2300 nM T66925 CML61O 10309583 IC50 = 700 nM T66925 C6JX2Q 11213817 IC50 = 420 nM T66925 C6B7PC 11379445 IC50 = 11000 nM T66925 CDA3Z4 11430157 IC50 = 170000 nM T66925 C3QD2E 11453435 IC50 = 110 nM T66925 CGYM83 43405474 IC50 = 770 nM T66925 CB15SK 44177708 IC50 > 50000 nM T66925 CF8R4L 44589634 IC50 > 200000 nM T66925 C5KSW0 44589636 IC50 = 5000 nM T66925 CZ3LE4 44590162 IC50 > 200000 nM T66925 C9H5JS 51039927 IC50 = 180 nM T66925 CHT9R4 52938041 IC50 = 320 nM T66925 C0ON6R 52938045 IC50 = 240 nM T66925 C9H5GZ 52938046 IC50 = 300 nM T66925 CEV19T 52938170 IC50 = 570 nM T66925 CF59EP 52938291 IC50 = 1200 nM T66925 C08STG 52938293 IC50 = 1300 nM T66925 C6YOG9 52938294 IC50 = 980 nM T66925 CY5VE4 52938668 IC50 = 310 nM T66925 CH9X0Y 52938669 IC50 = 280 nM T66925 C3ELI5 52938797 IC50 = 310 nM T66925 CVH6P1 52939047 IC50 = 1600 nM T66925 CW4A3I 52939048 IC50 = 600 nM T66925 C9G3TL 52939163 IC50 = 670 nM T66925 CMU46C 52939516 IC50 = 420 nM T66925 C4OK5Z 52939517 IC50 = 350 nM T66925 CNJ3E5 52939518 IC50 = 670 nM T66925 CM0B1P 52939519 IC50 = 430 nM T66925 CL1C8U 52939520 IC50 = 480 nM T66925 CV67SO 52939643 IC50 = 310 nM T66925 C4NY5P 52939644 IC50 = 250 nM T66925 C7X1PB 52939647 IC50 = 410 nM T66925 CHGK38 52939771 IC50 = 39 nM T66925 C0F5JG 52939772 IC50 = 850 nM T66925 CLF5S8 52939773 IC50 = 520 nM T66925 C3H8EG 52939774 IC50 = 440 nM T66925 CG49TO 52939776 IC50 = 340 nM T66925 CTCF48 52939902 IC50 = 960 nM T66925 C5HA4R 56953730 IC50 = 1100 nM T66925 CHNG07 56953735 IC50 = 500 nM T66925 C3Z8BE 56953736 IC50 = 340 nM T66925 CHYL72 56953863 IC50 = 220 nM T66925 C8AY9P 56953864 IC50 = 250 nM T66925 CI6L1M 56953865 IC50 = 570 nM T66925 CB4T3M 56953866 IC50 = 370 nM T66925 CJ4CU6 56953867 IC50 = 1400 nM T66925 C14JIX 56953989 IC50 = 500 nM T66925 C3WZA9 56953990 IC50 = 720 nM T66925 C19DEA 56954113 IC50 = 330 nM T66925 C3Q1MG 56954114 IC50 = 500 nM T66925 CZQ09H 56954116 IC50 = 230 nM T66925 CIAL27 56954117 IC50 = 380 nM T66925 CO7WI3 56954118 IC50 = 720 nM T66925 CJ9Z8T 56954217 IC50 = 310 nM T66925 CQP53N 56954218 IC50 = 280 nM T66925 CYV7I4 56954219 IC50 = 330 nM T66925 CF0L3O 56954220 IC50 = 760 nM T66925 CCS1W8 56954302 IC50 = 200 nM T66925 CNL06J 56954305 IC50 = 1500 nM T66925 CX89IJ 56954306 IC50 = 2200 nM T66925 CYB8K2 56954307 IC50 = 3300 nM T66925 C7RS2X 56954413 IC50 > 80000 nM T66925 C8HKW1 56954414 IC50 = 2500 nM T66925 CV2M0I 56954417 IC50 = 8900 nM T66925 CQ9G1B 56954418 IC50 > 80000 nM T66925 CQ06DB 56954502 IC50 > 80000 nM T66925 CK2W7N 56954503 IC50 = 27000 nM T66925 C9L3UE 56954504 IC50 > 80000 nM T66925 CJZ47H 56954507 IC50 = 870 nM T66925 CX3NW5 56954720 IC50 = 6700 nM T66925 C74KPC 56954722 IC50 = 6800 nM T66925 CL2B8Y 56954825 IC50 > 80000 nM T66925 C8XMJ9 56954826 IC50 = 16000 nM T66925 CZL5M6 56954827 IC50 = 740 nM T66925 CHA2O7 56954828 IC50 = 210 nM T66925 C3KSN7 56954829 IC50 = 51 nM T66925 CXQG95 56954830 IC50 = 66 nM T66925 C27JWY 56954942 IC50 = 180 nM T66925 C02CZV 58435684 IC50 > 100000 nM T66925 C1M7WL 70687120 IC50 = 2100 nM T66925 CNY61X 70688957 IC50 = 630 nM T66925 C4ZB7K 70693195 IC50 = 470 nM T66925 C1K5WF 70695295 IC50 > 26000 nM T66925 CDS6T7 71096277 IC50 > 50000 nM T66925 CWL96G 71449433 IC50 = 3600 nM T66925 CR9CK8 71450343 IC50 > 80000 nM T66925 C24YSA 71455725 IC50 = 21000 nM T66925 CB64IG 71456565 IC50 = 6400 nM T66925 CGM68H 71462877 IC50 = 35000 nM T66925 C62KMF 72204717 IC50 = 2000 nM T66925 CN6D1U 72204898 IC50 = 50000 nM T66925 CG0MH1 72204900 IC50 > 200000 nM T66925 CPN93S 72204902 IC50 > 200000 nM T66925 CIN2X8 72204904 IC50 = 30000 nM T66925 C7P2VY 72205081 IC50 > 200000 nM T66925 C1R6BL 72205083 IC50 > 200000 nM T66925 CI3PV6 72205085 IC50 > 200000 nM T66925 CJA86H 72205087 IC50 > 200000 nM T66925 C8WSG4 72205270 IC50 = 10000 nM T66925 CN52BD 72205272 IC50 = 20000 nM T66925 C93THM 72205274 IC50 > 200000 nM T66925 CYX2V6 76447116 IC50 = 46000 nM T66925 CF16UY 118722679 IC50 = 1700 nM T66925 CEAP41 118722680 IC50 = 1900 nM T66925 CD7I3Y 118722681 IC50 = 2200 nM T66925 C3INA2 118736260 IC50 = 220 nM T66925 CNQ12A 118736261 IC50 = 55 nM T66925 CW61EZ 118736262 IC50 = 48 nM T66925 CRT3P7 118736263 IC50 = 4 nM T66925 C7G1DH 118736264 IC50 = 720 nM T66925 C0Z8VF 118736265 IC50 = 130 nM T66925 C1BQM5 118736266 IC50 = 4 nM T66925 CX2Y0R 118736267 IC50 = 110 nM T66925 C02SAE 118736268 IC50 = 90 nM T66925 CL1O4F 118736269 IC50 = 430 nM T66925 CF32KR 118736270 IC50 = 86 nM T66925 CGK5M6 118736271 IC50 = 100 nM T66925 C5QM1T 136233424 IC50 > 80000 nM T21945 D00MYQ 4976 IC50 = 1.1 nM T21945 D00TLN 2913 Ki = 290 nM T21945 D01AXB 60835 IC50 = 4 nM T21945 D01JMC 11658860 Ki > 10000 nM T21945 D01UTL 2995 Ki = 0.6 nM T21945 D02PPN 4158 IC50 = 61 nM T21945 D02XOK 6917779 IC50 = 40 nM T21945 D03KQF 4011 Ki = 12 nM T21945 D03SKR 2803 IC50 > 20000 nM T21945 D04CRN 54841 IC50 = 3 nM T21945 D04WFD 4543 Ki = 6.3 nM T21945 D04XPW 446220 Ki = 108 nM T21945 D05GKD 33741 IC50 = 3600 nM T21945 D06GDY 43815 Ki = 90 nM T21945 D06ZUK 3696 Ki = 16 nM T21945 D07HQC 4236 IC50 = 283600 nM T21945 D08VRO 3822 Ki > 10000 nM T21945 D09VGC 65833 IC50 = 5500 nM T21945 D0CQ0Z 33630 Ki = 588 nM T21945 D0D1AL 3559 Ki = 5500 nM T21945 D0E6YQ 1935 IC50 = 11000 nM T21945 D0H4JM 8969 IC50 > 20000 nM T21945 D0H8QL 4020 IC50 = 4.9 nM T21945 D0J5RN 9690109 IC50 = 170000 nM T21945 D0K0TC 68617 IC50 = 825 nM T21945 D0O3FG 125017 IC50 = 538 nM T21945 D0P1UX 5656 IC50 = 149 nM T21945 D0T3LF 5826 EC50 = 7.1 nM T21945 D0T7OW 681 IC50 = 6.63 nM T21945 D0TR5X 3386 Ki = 440 nM T21945 D0X4ZR 444 IC50 = 1450 nM T21945 D0Y5DO 2771 Ki = 6190 nM T21945 D0Y5UG 2160 Ki = 333 nM T21945 D0ZS8P 2801 IC50 = 64.6 nM T21945 D00WLO 3455 IC50 = 79 nM T21945 D03QIE 47953 IC50 = 55 nM T21945 D04PXS 11658655 Ki = 63.1 nM T21945 D07AHC 65650 IC50 = 6500 nM T21945 D0C6QQ 60691 IC50 = 430 nM T21945 D0F5NJ 1615 Ki = 398 nM T21945 D0J9PT 58212050 IC50 = 8.8 nM T21945 D0LI1C 44469321 IC50 > 10000 nM T21945 D0R2OU 25070031 Ki = 10000 nM T21945 D0WL3H 15983287 IC50 = 763 nM T21945 D00OWF 5280953 Ki = 3260 nM T21945 D01NJT 65856 Ki = 0.3 nM T21945 D06BPG 4528 Ki = 3.8 nM T21945 D08AWI 11430856 Ki > 2000 nM T21945 D0A5RD 9795056 IC50 = 100 nM T21945 D0G1RH 6918446 IC50 = 0.2 nM T21945 D0H9GQ 9795276 IC50 = 20 nM T21945 CAG0J1 5523 IC50 = 3861 nM T21945 CK9A6Z 9280 IC50 = 51 nM T21945 C5H9CN 9287 Ki = 642 nM T21945 CRU9X7 16458 Ki > 10000 nM T21945 C3VL1J 27694 Ki = 128900 nM T21945 CGU3Z5 42145 Ki = 35200 nM T21945 CQR7U2 44024 IC50 = 22 nM T21945 C6WDL7 49756 Ki = 6380 nM T21945 CU86VK 54459 IC50 > 20000 nM T21945 C0OST7 55993 Ki = 4 nM T21945 C6KXM1 62857 IC50 = 4410 nM T21945 C9E6LD 62923 IC50 = 2550 nM T21945 CU65WJ 65327 Ki = 0.8 nM T21945 CI6QK3 77250 Ki = 5530 nM T21945 C8X5YU 77251 Ki = 7320 nM T21945 C0O3IG 77252 Ki = 3460 nM T21945 CYKE31 104920 IC50 = 1460 nM T21945 C5Q1OD 108220 Ki = 32.77 nM T21945 C3ZFS8 122252 Ki = 20 nM T21945 C3FW1L 132499 Ki = 125 nM T21945 CXUG79 148883 IC50 > 10000 nM T21945 CGT8R0 160510 Ki > 10000 nM T21945 CD1H4C 204666 IC50 = 2.8 nM T21945 CQ97NL 242919 Ki = 393 nM T21945 C1KUD9 264388 Ki > 10000 nM T21945 CR7MP9 264389 Ki > 10000 nM T21945 CDR63W 403508 Ki = 5.2 nM T21945 CYV1R3 417052 Ki > 4100 nM T21945 CZ53QF 656832 Ki = 1990 nM T21945 CZN6S9 743974 IC50 > 100000 nM T21945 C2CT0Y 818024 Ki = 230 nM T21945 CK65MQ 826771 IC50 = 2000 nM T21945 CH24PD 2801930 Ki = 37.52 nM T21945 CA3S7R 3022645 Ki = 1.1 nM T21945 CK8F0T 3080846 IC50 = 480 nM T21945 C9HJ3S 3302814 Ki = 1205 nM T21945 CJ6D8N 3342390 Ki < 1000 nM T21945 C0YXV3 3676358 Ki > 10000 nM T21945 CF12IO 4141883 Ki = 238 nM T21945 C9ZMC4 4476324 Ki = 2757 nM T21945 COC2V5 4913097 IC50 = 600 nM T21945 CI56AJ 5141361 Ki = 7.5 nM T21945 C5FUA2 6328322 Ki = 36300 nM T21945 C8ZK1O 6328354 Ki = 44 nM T21945 C0IHP9 6336338 Ki = 1.82 nM T21945 C2ICW4 9794964 Ki = 19 nM T21945 CDEL49 9795462 Ki = 47 nM T21945 C6XYV0 9795623 IC50 = 61 nM T21945 CR2JV1 9795977 Ki = 9 nM T21945 C5FJ4K 9798438 IC50 = 410 nM T21945 C7PUZ1 9816962 Ki = 5.8 nM T21945 CT7OD0 9817610 Ki = 8 nM T21945 CB8N5S 9817852 IC50 = 52 nM T21945 CEPW14 9834659 IC50 > 100000 nM T21945 CQPO85 9835750 Ki = 3.1 nM T21945 CX8P7C 9837869 Ki = 54 nM T21945 CY7K5Z 9838051 Ki = 12.3 nM T21945 C1YLP0 9838350 Ki = 5 nM T21945 C0YI3N 9839972 IC50 = 120 nM T21945 CM13ZV 9856041 Ki > 30000 nM T21945 CIXO17 9863396 IC50 = 10 nM T21945 C0IR5C 9864943 Ki = 96.7 nM T21945 C1ZB4W 9865652 Ki = 234 nM T21945 C3KGX7 9867350 Ki = 3.2 nM T21945 CN9YD5 9868131 IC50 = 200 nM T21945 CQ4LC2 9872676 Ki = 5090 nM T21945 CEJP40 9878793 IC50 = 275 nM T21945 C01ABG 9881528 Ki = 13.5 nM T21945 CLSP49 9881709 IC50 = 525 nM T21945 CCZ84V 9881969 Ki = 14 nM T21945 CT6C5H 9881970 Ki = 37 nM T21945 CHNC28 9882029 Ki = 13 nM T21945 CY6QX4 9882047 Ki = 7.2 nM T21945 C7KP4G 9882069 Ki = 19687 nM T21945 C8Q4OZ 9884474 Ki = 21 nM T21945 CBQ7Y3 9886288 Ki = 20 nM T21945 CN52BU 9887951 IC50 = 2700 nM T21945 CM3L0I 9900725 IC50 = 109 nM T21945 CCFR97 9903806 IC50 = 45 nM T21945 CPH07N 9903956 Ki = 16.5 nM T21945 CYWQ50 9906447 Ki > 10000 nM T21945 CUEZ75 9908121 Ki = 32 nM T21945 CCM2Z0 9908126 IC50 = 770 nM T21945 C1CSK2 9910220 IC50 = 1728 nM T21945 CSKJ62 9910492 IC50 = 540 nM T21945 C5T7UK 9921294 IC50 = 7100 nM T21945 C9MDU2 9921865 IC50 = 7400 nM T21945 CQX6R9 9924713 IC50 = 4200 nM T21945 C3RVK7 9928961 IC50 = 440 nM T21945 C10VOI 9930235 IC50 = 1000 nM T21945 CPYN79 9930791 IC50 = 1250 nM T21945 C6AZ3X 9943908 IC50 = 241 nM T21945 CPBQ94 9948049 IC50 = 200 nM T21945 C76NBU 9950374 Ki = 35 nM T21945 C5JI4O 9951619 IC50 = 270 nM T21945 CMI58L 9956563 IC50 = 0.037 nM T21945 CY9Q2M 9966187 IC50 = 17000 nM T21945 C7ZK5J 9966516 IC50 > 100000 nM T21945 CFZ9D7 9972515 IC50 = 1.1 nM T21945 COP08X 9972881 IC50 = 122 nM T21945 CXCP15 9980795 IC50 = 299 nM T21945 CQG25B 9993136 IC50 = 8200 nM T21945 C2AW8E 9996581 Ki = 5 nM T21945 CJ95XF 10003490 Ki = 29 nM T21945 CQL12P 10004545 Ki > 2000 nM T21945 CD9JO4 10015148 IC50 = 510 nM T21945 CHG91I 10017115 Ki = 663.8 nM T21945 CG6L4U 10042207 Ki > 8000 nM T21945 C25WVJ 10047566 IC50 > 1000 nM T21945 C5MQ9L 10060174 IC50 = 2.2 nM T21945 COZ94V 10062443 Ki = 269 nM T21945 C79GJK 10062560 Ki = 370 nM T21945 C1J4YU 10072978 Ki = 110 nM T21945 C1LN4V 10084648 Ki = 61 nM T21945 CO50KM 10085525 Ki = 1992 nM T21945 CW7K1U 10086952 Ki = 4720 nM T21945 C5H3MJ 10090352 IC50 = 6.9 nM T21945 CO1R2Q 10110820 IC50 = 770 nM T21945 CINW17 10130931 Ki = 35 nM T21945 C13VPI 10198613 Ki = 100 nM T21945 CM9CT0 10198980 Ki = 7.6 nM T21945 C4J6DM 10199240 Ki = 7.3 nM T21945 CF9B2N 10220613 Ki = 15 nM T21945 CG32IU 10220615 Ki = 135 nM T21945 CI8NQ2 10220697 Ki = 4.4 nM T21945 C8C6IY 10221010 IC50 = 7900 nM T21945 CYAV42 10236153 Ki = 10000 nM T21945 C6HUY5 10238982 Ki = 48.5 nM T21945 C2D4YM 10244152 IC50 > 100 nM T21945 CMSE68 10245407 IC50 = 11 nM T21945 CQ4M3F 10265481 Ki = 141.7 nM T21945 CNW1L9 10265758 IC50 = 121 nM T21945 C5AX7N 10291757 Ki = 184 nM T21945 C5HI6T 10293752 IC50 > 10000 nM T21945 CB4C9E 10313840 Ki = 219 nM T21945 C1Z8AO 10314993 Ki = 46 nM T21945 CKE53N 10320283 IC50 = 2210 nM T21945 CUF4G8 10355130 Ki = 28 nM T21945 CK1X4I 10356972 IC50 = 4 nM T21945 C4X6PO 10361811 Ki = 61 nM T21945 CRZ15J 10363398 Ki = 15 nM T21945 C3R7VI 10367506 IC50 = 93 nM T21945 CN1L4S 10377587 IC50 = 3700 nM T21945 CX13CN 10381502 Ki = 18 nM T21945 CRPS23 10399917 IC50 = 2300 nM T21945 CN2O8Q 10400315 Ki = 4.95 nM T21945 CUGW61 10403428 Ki = 21 nM T21945 C23LGF 10411109 Ki = 23 nM T21945 CI9ZQ8 10428183 IC50 = 23 nM T21945 CR8J7I 10432519 Ki > 1000 nM T21945 CRKC54 10439429 IC50 = 487 nM T21945 C98SIQ 10446567 Ki > 1000 nM T21945 CE5K4I 10447533 Ki = 26 nM T21945 CL65VJ 10450883 Ki = 242.29 nM T21945 CSZ56B 10472714 IC50 = 0.62 nM T21945 C1H3GU 10514152 IC50 > 20000 nM T21945 CF7B1H 10520686 Ki = 150 nM T21945 CX69HP 10525046 IC50 = 87 nM T21945 CJO95T 10537059 IC50 = 12800 nM T21945 CLOK62 10542372 IC50 = 13000 nM T21945 C7TX6Q 10543664 Ki = 2400 nM T21945 CJ6P1Z 10544672 Ki = 400 nM T21945 C3DR1F 10551367 Ki = 190 nM T21945 CRS7C2 10565247 IC50 > 20000 nM T21945 C0US7T 10568696 Ki = 650 nM T21945 C4U6NW 10575012 IC50 = 192 nM T21945 C3CYF7 10575547 IC50 > 10 nM T21945 CT1D8I 10586798 IC50 = 670 nM T21945 CC12NB 10591764 Ki = 75 nM T21945 CAGB14 10598649 Ki = 120 nM T21945 CN9RY5 10608447 IC50 > 20000 nM T21945 CQW4H8 10627068 Ki = 261 nM T21945 C6IQ0P 10635585 IC50 > 30000 nM T21945 CY3VA6 10636193 IC50 = 750 nM T21945 C8L4AG 10640435 Ki = 260 nM T21945 C69FME 10640436 Ki = 540 nM T21945 CCZU47 10663468 Ki = 150 nM T21945 C2P5WV 10666153 Ki = 855 nM T21945 CQ7V9F 10670209 IC50 > 10 nM T21945 CX12VM 10670307 Ki = 30 nM T21945 C9AW6Q 10685053 IC50 = 12000 nM T21945 C5FY3Q 10688125 Ki = 1100 nM T21945 CU58VP 10691286 Ki = 1600 nM T21945 CRLX06 10697639 Ki = 20 nM T21945 CV1I5H 10708388 IC50 = 2600 nM T21945 C54MCE 10711464 IC50 = 2600 nM T21945 C26VWI 10712698 Ki = 440 nM T21945 CB38TM 10727154 IC50 > 20000 nM T21945 CS7H2T 10729495 IC50 = 1400 nM T21945 C5Y6OZ 10729598 IC50 = 9900 nM T21945 CY39ZH 10731528 IC50 = 570 nM T21945 CPO3J8 10734429 Ki = 1500 nM T21945 C3I7ZE 10740824 IC50 = 279 nM T21945 CDZT46 10741033 Ki > 500 nM T21945 CR9U8L 10755592 IC50 = 1900 nM T21945 CRP3D6 10765459 IC50 = 205 nM T21945 C25OLB 10776648 IC50 > 20000 nM T21945 C3VXM8 10777680 IC50 = 1400 nM T21945 CP1N4Y 10788455 IC50 = 399 nM T21945 CGM3Q2 10788465 Ki = 82 nM T21945 CIC3J6 10799122 IC50 = 3600 nM T21945 CC12VQ 10800807 IC50 = 1400 nM T21945 CMN47B 10804265 IC50 = 2400 nM T21945 C2Q4BI 10813108 Ki = 41 nM T21945 CNB26G 10813109 Ki = 42 nM T21945 C9M7UN 10835740 Ki = 194 nM T21945 C0GX8V 10836499 Ki = 79 nM T21945 C1GAE4 10837110 Ki = 150 nM T21945 CZB85A 10850295 IC50 = 2200 nM T21945 CH40SM 10851277 IC50 = 3300 nM T21945 CAM8P0 10852732 IC50 = 44 nM T21945 C5JU4D 10860718 Ki = 690 nM T21945 CMS0Z2 10893018 Ki = 33.4 nM T21945 C58SAQ 10904197 Ki = 5.3 nM T21945 CE9JL7 10934835 IC50 = 1.9 nM T21945 C9VH4C 10946580 Ki = 191 nM T21945 CJC9K4 11005810 IC50 = 1140 nM T21945 CW0B4J 11034392 IC50 = 1.73 nM T21945 CEK01S 11044358 IC50 > 100000 nM T21945 CZ35QF 11045269 IC50 = 1.46 nM T21945 CFJG64 11059058 IC50 = 3020 nM T21945 C3XW2P 11077246 IC50 = 4.1 nM T21945 CIL61D 11077445 Ki = 11 nM T21945 C9KZ6L 11091998 IC50 = 260 nM T21945 C2ALP4 11130459 Ki = 0.9 nM T21945 CR6J8C 11130848 IC50 = 4.7 nM T21945 C36VJK 11149970 Ki = 7552 nM T21945 CT7Z9R 11150712 Ki = 0.3 nM T21945 C39INR 11150726 IC50 = 21 nM T21945 CP7O3X 11161917 Ki = 3823 nM T21945 CK27CU 11164446 Ki = 17 nM T21945 C7OEX0 11174494 Ki = 50 nM T21945 CLE8G5 11176087 Ki = 286 nM T21945 CAN73X 11189693 IC50 = 500 nM T21945 CM1T4L 11197267 IC50 = 93 nM T21945 CXQ48K 11198677 IC50 = 95 nM T21945 CPX23W 11209208 IC50 = 263 nM T21945 CPH9Q8 11210071 IC50 = 18000 nM T21945 C3VT2W 11219249 IC50 = 7.6 nM T21945 CCR0V5 11224454 Ki = 3910 nM T21945 CA39QR 11227406 Ki = 950 nM T21945 CR7IZ6 11231488 IC50 = 18.5 nM T21945 CQ7YK3 11244194 Ki = 717 nM T21945 CPVA01 11255359 IC50 = 11 nM T21945 C6IRX4 11265803 Ki = 483.55 nM T21945 CG4R6Y 11266831 Ki = 3 nM T21945 C6A0RY 11276613 Ki = 4440 nM T21945 C27GXZ 11277680 IC50 = 317 nM T21945 CZ86QW 11278193 Ki = 1034 nM T21945 CXH8G3 11278436 IC50 = 0.5 nM T21945 CV5F0G 11278895 IC50 = 100 nM T21945 CG9TM7 11293593 Ki = 7036 nM T21945 C57GTA 11299968 IC50 = 235 nM T21945 CP26RV 11300496 Ki = 135 nM T21945 C3F7NY 11301501 IC50 = 5700 nM T21945 CKQ7E8 11301538 Ki = 108 nM T21945 CV1LG4 11301893 IC50 = 9 nM T21945 CP12MY 11302314 IC50 = 57 nM T21945 CY26DK 11303722 Ki = 91 nM T21945 CS3BL0 11310988 Ki = 4600 nM T21945 CUXZ91 11311148 IC50 = 11.3 nM T21945 C2GZD3 11311204 IC50 = 86.7 nM T21945 CCJA60 11323414 Ki = 69 nM T21945 C2FK4V 11325961 IC50 = 225 nM T21945 CBA4U5 11335494 IC50 = 24.9 nM T21945 CF2X6Y 11336016 Ki = 37 nM T21945 CH83FN 11346324 Ki = 445.36 nM T21945 CXZ82E 11347860 Ki = 17 nM T21945 C3O0EP 11349976 Ki = 214 nM T21945 C4ZP2J 11358065 IC50 = 290 nM T21945 CR5S4A 11368527 IC50 = 88 nM T21945 C7MN8V 11391287 IC50 = 18 nM T21945 CE85CL 11415039 IC50 = 22.8 nM T21945 CE2TS1 11425104 Ki > 10000 nM T21945 CU4H7W 11426687 Ki = 4332 nM T21945 C9QPU4 11427925 IC50 = 255 nM T21945 C85LYP 11430418 IC50 > 1000 nM T21945 CSJ87M 11438393 Ki = 160.8 nM T21945 C6E3VO 11449834 IC50 = 800 nM T21945 C3TK6Z 11450294 IC50 = 720 nM T21945 CMH9J5 11450298 IC50 = 5 nM T21945 CX3ZU0 11450539 IC50 = 12 nM T21945 C10WNZ 11450786 IC50 = 550 nM T21945 CNS8J9 11459667 IC50 = 12.4 nM T21945 CZAV70 11463320 Ki = 417 nM T21945 CF5R1Z 11463970 IC50 = 26 nM T21945 C9L2AH 11474847 IC50 = 310 nM T21945 C2X3OY 11483535 Ki = 946.2 nM T21945 C4XC1L 11485581 Ki = 140 nM T21945 CZ7X9M 11492164 Ki = 8517 nM T21945 C7G5HP 11492305 IC50 > 10000 nM T21945 CA8KE0 11492902 IC50 = 8900 nM T21945 C3XD4T 11493035 Ki > 10000 nM T21945 C2NJY3 11499666 IC50 = 3392 nM T21945 C2X7HI 11499753 Ki > 10000 nM T21945 C7UJM8 11499957 IC50 = 120 nM T21945 CDC5I4 11499958 Ki = 23 nM T21945 CXR70Z 11500795 Ki = 1120 nM T21945 CIN4B7 11500848 IC50 = 62 nM T21945 C3B0LO 11501191 Ki = 7 nM T21945 CR1K9A 11504964 Ki = 40 nM T21945 C2Y0JA 11505593 Ki = 402 nM T21945 CS1YI5 11506975 IC50 > 10000 nM T21945 C9OV2L 11507416 IC50 = 52 nM T21945 C6FA1G 11513575 Ki = 91 nM T21945 CM3P5D 11514441 Ki > 10000 nM T21945 C4DB0Z 11515426 IC50 = 70 nM T21945 C9XYF3 11521964 IC50 = 350 nM T21945 C75FPD 11529874 Ki = 6 nM T21945 C3IBX7 11529992 IC50 = 31 nM T21945 C38QFE 11530118 Ki > 10000 nM T21945 C6SCW7 11536158 Ki = 455 nM T21945 CDM6F9 11536862 Ki = 30 nM T21945 CC67XR 11543737 IC50 = 224 nM T21945 CGV24I 11544186 IC50 = 37 nM T21945 CWCU85 11548538 Ki = 143 nM T21945 CTXP63 11550888 IC50 = 130 nM T21945 C9VC7O 11551780 Ki > 10000 nM T21945 C51PVS 11558708 IC50 = 31 nM T21945 C3RMI1 11559300 Ki = 9 nM T21945 CY71DQ 11562044 Ki = 79 nM T21945 CH9MP0 11566229 Ki = 30 nM T21945 C1VF0P 11566266 Ki = 8 nM T21945 CDP9Z0 11566316 Ki = 8 nM T21945 C8C1VW 11566318 Ki = 9 nM T21945 CIE3O7 11566487 Ki > 10000 nM T21945 CZD62R 11572546 IC50 = 726 nM T21945 CMX60P 11573849 IC50 = 16 nM T21945 C6JC2T 11580039 Ki > 10000 nM T21945 CD5XT0 11580456 IC50 = 25 nM T21945 C2T6RF 11584839 Ki = 103 nM T21945 CMZ54K 11587069 IC50 = 481 nM T21945 C3LAI9 11587242 IC50 = 6.8 nM T21945 CY3A4K 11587772 Ki = 5 nM T21945 CU8F6B 11588595 IC50 = 110 nM T21945 CI12ZR 11592176 Ki = 43 nM T21945 CW1CO6 11594137 IC50 = 22 nM T21945 CZ6US0 11594677 IC50 = 19.3 nM T21945 CJ27XH 11594827 Ki = 0.76 nM T21945 CAD20M 11598831 Ki = 485 nM T21945 C9YR3G 11599258 Ki = 359 nM T21945 C7UFA1 11600778 IC50 > 10000 nM T21945 C6YB7K 11602095 Ki = 63 nM T21945 CE4GZ0 11609767 IC50 = 2520 nM T21945 C6HLN8 11610150 Ki = 3 nM T21945 C8JAM4 11616357 IC50 = 1300 nM T21945 CCM6U9 11616771 Ki = 25 nM T21945 C1F4DL 11618807 Ki = 118 nM T21945 CI2VM7 11620991 Ki = 440 nM T21945 C5FQR2 11622909 IC50 = 0.7943 nM T21945 C4YI2U 11623560 IC50 = 98 nM T21945 C1KD4Z 11623823 IC50 = 28 nM T21945 C86SZO 11624458 IC50 = 29 nM T21945 CYEH35 11627756 Ki = 785 nM T21945 C0I1YV 11628203 Ki = 560 nM T21945 CA8IM9 11630375 Ki = 110 nM T21945 CF0QR8 11630988 Ki = 10 nM T21945 CXJ73O 11638552 Ki = 36 nM T21945 CQ1U9W 11638962 Ki = 6 nM T21945 C3VOG6 11644931 IC50 = 3360 nM T21945 C97OLY 11649733 Ki = 361 nM T21945 CX2ZD7 11650267 IC50 = 957 nM T21945 C7BM5S 11650367 Ki = 338 nM T21945 C3OC6J 11650990 Ki = 177 nM T21945 CL4AJ0 11658719 IC50 = 2126 nM T21945 CAZN26 11659436 IC50 = 60 nM T21945 CF92SM 11659664 IC50 = 23 nM T21945 C0KH7D 11660186 IC50 = 39 nM T21945 CIX54K 11666319 IC50 = 19 nM T21945 C1SYE2 11667017 IC50 = 64 nM T21945 CJ9Z8D 11671232 Ki = 160 nM T21945 C98NXK 11671382 Ki = 736 nM T21945 C8Q5WO 11674313 Ki = 6.8 nM T21945 CT3BP5 11674529 Ki = 95 nM T21945 C79PHA 11678447 Ki = 330 nM T21945 C5Q3ZU 11680542 Ki = 63.1 nM T21945 C2DBG7 11687579 IC50 = 13 nM T21945 C0Y6OR 11687843 Ki = 74 nM T21945 C8R7TP 11694495 IC50 = 374 nM T21945 C6T8ZD 11694789 IC50 = 7.8 nM T21945 CL19UR 11701869 IC50 = 10 nM T21945 CYN4H9 11702602 Ki = 5 nM T21945 C5OZD6 11706276 Ki > 5600 nM T21945 CZB5P9 11709831 Ki = 34 nM T21945 C4M9AU 11710505 Ki = 13 nM T21945 CQWL60 11713341 Ki = 210 nM T21945 C18ZHK 11713731 Ki = 947 nM T21945 CHRM03 11716290 IC50 = 4715 nM T21945 CKQ03I 11716308 Ki = 634 nM T21945 CN2L4J 11716660 IC50 = 3.4 nM T21945 C5BQV8 11723540 IC50 = 240 nM T21945 C4MC2V 11740717 Ki = 699 nM T21945 C2QZI5 11771101 Ki = 194 nM T21945 CN4Y8B 11778700 IC50 = 18 nM T21945 CKNE31 11791987 Ki = 2200 nM T21945 CW15BI 11794260 Ki > 10000 nM T21945 CN9M8E 11811722 IC50 = 2810 nM T21945 CJO0Q6 11818515 Ki > 10000 nM T21945 C2UT9D 11846746 IC50 = 754 nM T21945 CRX17H 11855337 Ki = 21 nM T21945 CXLW54 11948707 Ki > 10000 nM T21945 C8EJ6H 11949672 IC50 = 8 nM T21945 CK13QD 11953409 Ki = 7700 nM T21945 C8JQL7 11957735 IC50 > 10000 nM T21945 C5QB3M 11963972 IC50 = 30 nM T21945 CAW2Y1 12000105 Ki = 4168 nM T21945 C49HJG 12122109 Ki = 0.95 nM T21945 CUFP52 12149037 IC50 = 161 nM T21945 CT4RA6 12204576 IC50 = 4.9 nM T21945 CK6WG1 12276477 IC50 = 5761 nM T21945 C2MP5H 12559279 IC50 > 10000 nM T21945 C6MH2K 12646716 IC50 = 158000 nM T21945 CYU4P5 12739458 Ki > 10000 nM T21945 C0KR1M 12884652 Ki = 1200 nM T21945 CM78FI 12999584 IC50 = 128 nM T21945 CCG14E 13091356 Ki = 1791 nM T21945 CYN95Z 13091359 Ki = 1409 nM T21945 C9CF3W 13520310 IC50 = 120 nM T21945 C1FAP2 13520317 IC50 = 208 nM T21945 CQV86I 13718739 IC50 > 10000 nM T21945 CGY6Q3 13718746 IC50 = 2800 nM T21945 C0KU4R 13718753 IC50 = 3700 nM T21945 C12NSL 13718761 IC50 = 6500 nM T21945 CI6TP9 13903189 Ki = 16.6 nM T21945 CHJ27K 13903191 Ki = 4.1 nM T21945 C4KU1J 14014888 IC50 > 10000 nM T21945 CO7N1M 14422827 IC50 = 4700 nM T21945 CQI9F6 14571114 Ki = 137 nM T21945 CFZP25 14601687 IC50 = 6200 nM T21945 C9GEN5 14674210 IC50 > 10000 nM T21945 C8UBJ4 15015316 Ki = 55 nM T21945 CJ8WL9 15015330 Ki = 20 nM T21945 C0P5LY 15069893 Ki = 1110 nM T21945 CE4T7Z 15069894 Ki = 39 nM T21945 C8SXL1 15069905 Ki = 23 nM T21945 CMI6C8 15113388 Ki = 31.8 nM T21945 C27ZJA 15113390 Ki = 1020 nM T21945 CD24IR 15115364 IC50 = 3100 nM T21945 CTZ61G 15132121 IC50 = 50 nM T21945 C2T1UK 15290836 IC50 = 57 nM T21945 CO6P8K 15405849 IC50 = 2.2 nM T21945 C53JMI 15639786 Ki = 10 nM T21945 C1FLJ0 15639787 Ki = 19 nM T21945 C4OT1S 15639792 Ki = 458 nM T21945 CM2UZ3 15949838 Ki = 156 nM T21945 C2ZYA6 15951338 IC50 = 400 nM T21945 CL0SF3 15951408 IC50 = 160 nM T21945 C1Q8IV 15951410 IC50 = 380 nM T21945 CW8M6S 15952123 IC50 = 770 nM T21945 CM6O3G 15983286 IC50 = 644 nM T21945 C89XFJ 16007138 Ki = 20 nM T21945 CG60DM 16038376 IC50 = 53 nM T21945 C37FIP 16047544 Ki = 2733 nM T21945 CL0B8J 16063251 IC50 = 91 nM T21945 CO58NM 16067544 IC50 > 3000 nM T21945 C4LFH6 16067545 IC50 > 3000 nM T21945 C5KHE3 16067546 IC50 = 26 nM T21945 CR8F9E 16067547 IC50 = 14 nM T21945 CE4A2K 16067549 IC50 > 3000 nM T21945 CJRU09 16067550 IC50 = 7 nM T21945 C8PL4S 16067551 IC50 = 175 nM T21945 CTS91K 16067641 IC50 = 44 nM T21945 CP54FR 16067643 IC50 = 166 nM T21945 CS81ZB 16067645 IC50 = 22 nM T21945 CPLR62 16067646 IC50 = 627 nM T21945 C0VK4Y 16067647 IC50 = 32 nM T21945 CQ4P2J 16067648 IC50 = 215 nM T21945 CAY61X 16067730 IC50 = 9 nM T21945 C7ZK3R 16067731 IC50 = 463 nM T21945 CV7XN9 16067732 IC50 = 201 nM T21945 CRD3S8 16067733 IC50 = 311 nM T21945 C3QMW5 16067734 IC50 = 121 nM T21945 CLY3X5 16067834 IC50 = 1053 nM T21945 C8I6EM 16067835 IC50 = 30 nM T21945 C83KQX 16067839 IC50 = 19 nM T21945 CJ24NE 16067840 IC50 = 6 nM T21945 C2RA5B 16067943 IC50 = 7 nM T21945 CTG78M 16067944 IC50 = 6 nM T21945 CR07MN 16067945 IC50 = 19 nM T21945 CEVD42 16091071 Ki = 2470 nM T21945 CH74RZ 16102752 IC50 = 51 nM T21945 C6OR3H 16102755 Ki = 830 nM T21945 C9SH0B 16102756 IC50 = 730 nM T21945 CA75KZ 16102757 IC50 = 730 nM T21945 C1L9HQ 16102758 IC50 = 1700 nM T21945 CMUI02 16102759 Ki = 2900 nM T21945 CLO54U 16102760 IC50 = 680 nM T21945 C3SEF2 16102761 Ki = 490 nM T21945 CYF03S 16102762 Ki = 970 nM T21945 C4N9BG 16102763 Ki = 380 nM T21945 C2HLF8 16102765 Ki = 12 nM T21945 CTX94E 16102766 IC50 = 9 nM T21945 C9HLB7 16102767 IC50 = 410 nM T21945 CLHY18 16102768 IC50 = 330 nM T21945 CG90ID 16102769 Ki = 2500 nM T21945 CH53XS 16102770 IC50 = 28 nM T21945 CJ32XS 16113210 IC50 = 100 nM T21945 C9UYE0 16126667 Ki = 257 nM T21945 C5ES3D 16126745 Ki = 10.8 nM T21945 C4QCP3 16494915 IC50 = 9987 nM T21945 C2VQS3 16640939 IC50 = 9200 nM T21945 C6P4BX 16656803 IC50 = 158 nM T21945 CZ2IS9 16660294 Ki > 10000 nM T21945 CW40DA 16678084 IC50 = 30 nM T21945 CH4Y2D 16681434 IC50 = 148 nM T21945 CDT5V8 16721129 Ki = 106 nM T21945 CL5G7A 16730754 Ki = 268 nM T21945 CUG5B8 16747689 Ki = 201 nM T21945 C50YME 16747877 IC50 = 912 nM T21945 CY8QO6 16748004 IC50 = 960 nM T21945 CY2FL4 16748005 IC50 = 582 nM T21945 C9CQ1B 16748006 IC50 = 620 nM T21945 COGJ31 16748007 IC50 = 1820 nM T21945 CPF2K0 16748165 Ki = 990 nM T21945 CM1L6Q 16748381 Ki = 1910 nM T21945 CG5FU0 16748382 Ki = 1630 nM T21945 CYN9W8 16748383 IC50 = 1550 nM T21945 CM89SX 16748512 IC50 = 1810 nM T21945 C1ZQX9 16748513 Ki = 1390 nM T21945 CM46NI 16748623 IC50 = 650 nM T21945 C9W7LH 16748731 Ki = 2210 nM T21945 CJ9S7I 16748848 IC50 = 690 nM T21945 CXH10U 16748849 IC50 = 2300 nM T21945 C37DZJ 16748949 Ki = 2300 nM T21945 CTJ2Z3 16748950 IC50 = 1170 nM T21945 C1L8DV 16748951 IC50 = 4000 nM T21945 CTI89R 16759249 Ki = 1330 nM T21945 CN4HB8 18391094 Ki = 550 nM T21945 CH39LP 18391096 Ki = 626 nM T21945 C03IZO 18623856 IC50 = 8.2 nM T21945 C9JD5Y 19360456 IC50 = 300 nM T21945 CO25RM 19857878 IC50 = 6900 nM T21945 CYFJ81 19926671 IC50 = 256 nM T21945 C21LXU 20055336 Ki = 130 nM T21945 C8ICF9 20111627 IC50 = 21 nM T21945 C6R8AM 20631904 Ki = 1.2 nM T21945 C81FRQ 20636465 Ki = 388 nM T21945 CXQM78 20695745 IC50 = 1570 nM T21945 CEO8W1 21116177 IC50 = 86 nM T21945 CVD6F9 21241523 Ki = 745 nM T21945 CRV56X 21365270 IC50 = 51 nM T21945 C3T5HF 21509921 Ki > 10000 nM T21945 CFN81Q 21527771 Ki = 3959 nM T21945 CH59WN 21533446 Ki = 2249 nM T21945 C9H4XW 21539375 IC50 = 3570 nM T21945 C27GSH 21539381 IC50 = 5176 nM T21945 C2X0TW 22337167 Ki = 39119 nM T21945 CR4T9J 22337182 Ki > 100000 nM T21945 CQUY92 22386812 Ki = 116 nM T21945 C7O8WZ 22386894 Ki = 8.8 nM T21945 CMDI47 22386922 Ki = 136 nM T21945 CW5M2S 22419110 Ki = 1039 nM T21945 CU8YV6 22468266 IC50 = 45 nM T21945 CF6P4V 22468271 Ki = 183 nM T21945 CV2XH0 22798952 IC50 = 562.34 nM T21945 CPH6L4 22966050 Ki = 1820 nM T21945 CYPV48 23378645 IC50 = 760 nM T21945 C4ATJ7 23378652 IC50 = 7900 nM T21945 C57EFO 23378743 IC50 = 6700 nM T21945 CL45FG 23519626 IC50 = 6688 nM T21945 CDJR16 23519628 IC50 = 1010 nM T21945 CF3SU0 23519629 IC50 = 3867 nM T21945 C7YFT3 23582127 Ki = 11 nM T21945 C57MTL 23625757 Ki = 96 nM T21945 C6IF2N 23661687 Ki > 100000 nM T21945 CSB9E8 24103136 IC50 = 640 nM T21945 CL4WV2 24180125 IC50 = 2470 nM T21945 C0I5RA 24180665 IC50 = 710 nM T21945 C91IVZ 24742317 IC50 = 9.4 nM T21945 C32IVO 24742475 IC50 = 5.8 nM T21945 CWGH86 24743352 IC50 = 21 nM T21945 CYBG40 24743354 IC50 = 20 nM T21945 CG3XD5 24743436 IC50 = 6.5 nM T21945 C61QPT 24748794 Ki = 11 nM T21945 C9P2NE 24748795 Ki = 7 nM T21945 CYRZ48 24749837 Ki = 37 nM T21945 C4Y0BF 24749952 Ki = 95 nM T21945 CJ2N8B 24749953 Ki = 14 nM T21945 CV30EH 24749955 Ki = 56 nM T21945 CPD4M8 24749956 Ki = 279 nM T21945 CO7TD4 24750311 Ki = 7.5 nM T21945 C4R9YO 24750312 Ki = 97 nM T21945 C60SIH 24750313 Ki = 114 nM T21945 C2ZJ3Q 24750421 Ki = 12 nM T21945 CV1K6O 24750422 Ki > 1000 nM T21945 CQ1G3S 24750423 Ki = 33 nM T21945 C16YHA 24764464 IC50 = 12 nM T21945 CHI83W 24769038 IC50 = 5.4 nM T21945 C5ASY1 24773552 Ki = 725 nM T21945 C1FIS5 24773804 Ki = 618 nM T21945 C9KXC8 24773805 Ki = 467 nM T21945 CP1F6M 24782241 Ki = 7.943 nM T21945 CZ2XE7 24782243 Ki = 501.19 nM T21945 CJQ2X4 24782485 Ki = 6.31 nM T21945 CI7S2G 24782486 Ki = 25.12 nM T21945 CK5TO1 24782487 Ki = 251.19 nM T21945 CZ34RN 24782489 Ki = 15.85 nM T21945 CL5GS1 24786064 Ki = 50.12 nM T21945 CQN4W1 24802843 Ki = 100 nM T21945 C23ICW 24802846 Ki = 100 nM T21945 CX6ZB7 24802848 Ki = 794.33 nM T21945 CH30VR 24803009 Ki = 199.53 nM T21945 CH87VD 24803010 Ki = 7.943 nM T21945 CC78ZE 24803012 Ki = 50.12 nM T21945 C7C4UQ 24803014 Ki = 199.53 nM T21945 C17ISZ 24803180 Ki = 3162.28 nM T21945 C4O8ZF 24803181 Ki = 125.89 nM T21945 C1W8NS 24803185 Ki = 316.23 nM T21945 C9LV3D 24803344 Ki = 79.43 nM T21945 C96CBA 24803345 Ki = 316.23 nM T21945 CWE46Z 24810003 Ki = 4790 nM T21945 C8TZY0 24810004 Ki = 2080 nM T21945 C85LUK 24822173 IC50 = 29 nM T21945 C0M7CN 24825720 Ki = 181.97 nM T21945 CDC91N 24839550 Ki = 1000 nM T21945 C1CUD0 24848444 Ki = 5920 nM T21945 C6ZRA7 24849533 Ki = 100 nM T21945 C50XIV 24855884 Ki = 140 nM T21945 CJTY89 24855886 Ki = 5700 nM T21945 C79FCO 24855918 Ki = 760 nM T21945 CJAC42 24855949 Ki = 470 nM T21945 C1SVD5 24855952 Ki = 3300 nM T21945 C0DUL3 24857666 IC50 = 124 nM T21945 CC8J1Z 24857667 IC50 = 731 nM T21945 C9V5MT 24857668 IC50 = 855 nM T21945 C5QGY4 24857669 IC50 = 174 nM T21945 CSR8J4 24857759 IC50 = 26 nM T21945 C27EUV 24857839 IC50 = 8.7 nM T21945 CZ8TA6 24857854 IC50 = 1.7 nM T21945 C97SEP 24857858 Ki = 1680 nM T21945 CBI5D7 24860769 IC50 = 3200 nM T21945 C7COU6 24860831 IC50 = 120 nM T21945 CVO64M 24860832 IC50 = 4000 nM T21945 CL26KS 24860835 IC50 = 330 nM T21945 C7EHG5 24860898 IC50 = 8733 nM T21945 C2X6VF 24860899 IC50 = 4000 nM T21945 CAU07P 24860900 IC50 > 10000 nM T21945 CM9L7D 24860902 IC50 = 2783 nM T21945 CZ3R7W 24860903 IC50 = 890 nM T21945 CG8T3J 24860904 IC50 = 170 nM T21945 CH2BO5 24861136 Ki = 45 nM T21945 CY18GS 24861188 Ki = 306 nM T21945 C70MST 24861189 Ki = 78 nM T21945 CW1NB6 24861190 IC50 = 302 nM T21945 CZ2OX1 24861191 Ki = 25 nM T21945 CA1VQ4 24861192 Ki = 428 nM T21945 C54HEN 24861246 Ki = 28 nM T21945 C2GPJ5 24861249 Ki = 73 nM T21945 CU90ZK 24861250 Ki = 27 nM T21945 CAK91U 24861356 IC50 = 116 nM T21945 CO51AG 24863961 Ki > 100000 nM T21945 CD9SF2 24863962 Ki > 100000 nM T21945 CXD45U 24867041 IC50 = 23 nM T21945 CV1PY2 24878951 Ki > 100000 nM T21945 CK6JC4 24878953 Ki > 100000 nM T21945 C4SL0V 24879001 Ki = 58100 nM T21945 C3Z4JN 24879003 Ki > 10000 nM T21945 C56IDA 24879005 Ki > 100000 nM T21945 C23LNY 24879008 Ki > 100000 nM T21945 C9C8OH 24879010 Ki > 100000 nM T21945 C1ZRH6 24879054 Ki > 10000 nM T21945 CD17RE 24879056 Ki > 10000 nM T21945 CX20BZ 24879058 Ki > 10000 nM T21945 C9A2NF 24890939 Ki = 3200 nM T21945 CG0Z8X 24893996 IC50 = 5600 nM T21945 CQH6A4 24894787 Ki = 1376 nM T21945 CJ8K0T 24894790 Ki = 1220 nM T21945 CMTK42 24894905 Ki = 117 nM T21945 CYKD83 24894907 Ki = 187 nM T21945 CH04XN 24894909 Ki = 785 nM T21945 CB51HT 24894913 Ki = 368 nM T21945 C46VNQ 24895014 Ki = 41 nM T21945 CV9E4X 24895015 IC50 = 303 nM T21945 C9YUR2 24895017 Ki = 519 nM T21945 CRN96X 24895020 Ki = 58 nM T21945 C3RH4A 24895022 Ki = 514 nM T21945 C1LX7D 24895129 Ki = 544 nM T21945 C0EYS5 24895131 Ki = 14 nM T21945 C8ER2O 24897032 IC50 = 68 nM T21945 C0Z4PW 24897264 IC50 = 156 nM T21945 C5HPS8 24897268 IC50 = 30 nM T21945 CT0HG9 24897269 IC50 = 217 nM T21945 CB37QM 24897270 IC50 = 61 nM T21945 C7B3YH 24897482 IC50 = 29 nM T21945 CMP23U 24897483 IC50 = 240 nM T21945 CQ1N4S 24897484 IC50 = 20 nM T21945 CN3XK4 24897486 IC50 = 23 nM T21945 CH1PU0 24897487 IC50 = 400 nM T21945 CNH7C9 24897687 IC50 = 73 nM T21945 C48GLF 24897688 IC50 = 110 nM T21945 CTG6D4 24897689 IC50 = 34 nM T21945 C4FEQ6 24936132 Ki = 1.21 nM T21945 CF2A7C 24936614 IC50 = 1 nM T21945 CLG21T 24937260 IC50 = 147 nM T21945 CR5F7V 24937375 IC50 = 2304 nM T21945 C61XEY 24937629 IC50 = 30 nM T21945 CTM10X 24937631 IC50 = 94 nM T21945 C4G8UV 24937633 IC50 = 4.5 nM T21945 C6I4YO 24937759 IC50 = 10 nM T21945 C94UGH 24937889 IC50 = 2 nM T21945 C5U9FD 24937892 IC50 = 57 nM T21945 C3H5PJ 24947569 Ki = 3700 nM T21945 C4Y7FP 24947750 Ki = 530 nM T21945 CA8VN2 24947751 Ki = 470 nM T21945 CYGT57 24947752 Ki = 730 nM T21945 CEW8C3 24947936 Ki = 2000 nM T21945 C6BIR1 24947941 Ki = 4800 nM T21945 C06TLI 24948121 Ki = 1300 nM T21945 CW4X0E 24962988 Ki = 8 nM T21945 CQ42YZ 24964158 Ki = 290 nM T21945 C4P5AD 24964159 Ki = 240 nM T21945 CB9C4E 24965063 Ki > 6000 nM T21945 CZXC58 24965064 Ki > 6000 nM T21945 CT39VO 24969452 IC50 = 8 nM T21945 CGZ60N 24969453 IC50 = 8 nM T21945 CKNQ63 25008443 IC50 = 2250 nM T21945 CZ6T5Q 25009937 Ki = 8 nM T21945 CQ9LS6 25022704 Ki = 10 nM T21945 C0HRL1 25024305 Ki = 19.95 nM T21945 C2RQX9 25024309 Ki = 100 nM T21945 C3W1NC 25024503 Ki = 251.19 nM T21945 CY0VU5 25025577 Ki = 223.87 nM T21945 CA20NZ 25025581 IC50 = 0.1585 nM T21945 CU8A6N 25025776 Ki = 0.631 nM T21945 C4I5LJ 25025778 Ki = 1.585 nM T21945 CPJD86 25025779 Ki = 0.631 nM T21945 CN0U3C 25025780 Ki = 15.85 nM T21945 CFAZ02 25025782 Ki = 0.3981 nM T21945 CDX2C6 25025977 Ki = 0.2512 nM T21945 CRQ73B 25025978 Ki = 1.259 nM T21945 C9WQ5K 25025979 Ki = 0.1585 nM T21945 C16YGB 25029543 IC50 = 130 nM T21945 CIBS51 25029544 IC50 = 630 nM T21945 CEFH96 25029545 IC50 = 1030 nM T21945 C8GC4E 25029546 IC50 = 790 nM T21945 CT3M0B 25029547 IC50 = 910 nM T21945 CF3X4K 25029548 IC50 = 1500 nM T21945 C9RSA0 25029788 IC50 = 490 nM T21945 CBQ48M 25029789 IC50 = 140 nM T21945 CI2O0G 25029790 IC50 = 3550 nM T21945 CIO09R 25029791 IC50 = 970 nM T21945 C5M0NJ 25029792 IC50 = 200 nM T21945 CZX10T 25030029 IC50 = 38 nM T21945 CZ7C0R 25030031 IC50 = 1400 nM T21945 CE89TZ 25030033 IC50 = 120 nM T21945 CZOR47 25030035 IC50 = 30 nM T21945 CA4L5Q 25032786 IC50 > 10 nM T21945 C6K4SH 25033519 IC50 = 11 nM T21945 CPT9X8 25066443 IC50 = 26 nM T21945 CIWT97 25071015 Ki = 102 nM T21945 CP9J7Q 25071019 IC50 = 4 nM T21945 CF3S2A 25109015 IC50 = 88 nM T21945 C9V8CQ 25109439 IC50 = 55 nM T21945 CR86IN 25109441 IC50 = 93 nM T21945 C82OWZ 25109445 IC50 = 52 nM T21945 C61LDS 25109651 IC50 = 170 nM T21945 CGBL04 25139014 Ki = 4490 nM T21945 CJ5VX0 25140466 Ki = 845 nM T21945 C0YEI8 25141192 Ki = 454 nM T21945 C0MPE3 25141372 Ki > 5200 nM T21945 C0OT1F 25141373 Ki > 1200 nM T21945 C7W9YX 25150535 IC50 = 15 nM T21945 C35XQI 25150621 IC50 = 2.3 nM T21945 CD0QU5 25150624 IC50 = 17 nM T21945 CIZ1N9 25150625 IC50 = 13 nM T21945 C6IXV9 25150627 IC50 = 19 nM T21945 CE1ND3 25150628 IC50 = 6 nM T21945 CAVR45 25150711 IC50 = 4.4 nM T21945 CW9MX8 25168440 Ki = 9 nM T21945 CXC35U 25168857 IC50 = 1.5 nM T21945 C30VBG 25181825 IC50 = 3200 nM T21945 C4W2AK 25181826 IC50 = 2000 nM T21945 C7JYI8 25188212 Ki = 3.14 nM T21945 C56CDP 25188770 Ki = 1.02 nM T21945 C5Z0LT 25188771 Ki = 3.68 nM T21945 C46ANM 25195291 Ki = 18 nM T21945 C37YTG 25210603 Ki = 2.512 nM T21945 CW3JR1 25210604 Ki = 25.12 nM T21945 CCTO39 25210872 Ki = 1.995 nM T21945 CE7BA0 25210873 Ki = 7.943 nM T21945 C0FE8U 25210874 Ki = 7.943 nM T21945 C0XN3L 25210876 Ki = 1.585 nM T21945 CF6AD3 25211583 Ki = 4600 nM T21945 CVU7J1 25211682 Ki = 6567 nM T21945 CC47VW 25253703 IC50 = 10.4 nM T21945 C76XYF 25253914 IC50 = 257 nM T21945 C49CDZ 25253915 IC50 = 36.7 nM T21945 CFI0K3 25253916 IC50 = 13.8 nM T21945 CG6C7H 25253917 IC50 = 4.1 nM T21945 CX07CK 25258806 Ki = 39119 nM T21945 CHY8S9 25258809 Ki = 19332 nM T21945 C3F0CJ 25260132 IC50 = 16 nM T21945 C7PK2X 29938807 Ki = 3.3 nM T21945 CSO5Y3 29981497 Ki = 97100 nM T21945 CN8J0W 29981513 Ki > 10000000 nM T21945 CJ1N0X 29981679 Ki = 920000 nM T21945 CH3M1E 31413243 IC50 > 10000 nM T21945 C9GS1N 31413320 IC50 > 10000 nM T21945 C2XY4V 31413484 IC50 > 10000 nM T21945 CW2KO7 31568498 IC50 = 6070 nM T21945 CHE3I4 33139722 IC50 > 10000 nM T21945 C4FR6G 36465568 IC50 > 10000 nM T21945 CRD0C3 42273320 IC50 = 4960 nM T21945 C2TUQ3 42273630 IC50 > 10000 nM T21945 C7C9DY 42629242 IC50 = 99 nM T21945 CRQ96D 42634153 IC50 = 280 nM T21945 C1J4XZ 42636222 IC50 = 1 nM T21945 CR70ZY 43164282 IC50 = 273 nM T21945 CNL52R 43283283 IC50 = 42 nM T21945 C6P5DK 43283415 IC50 = 22 nM T21945 C1YM3D 44131466 Ki = 276 nM T21945 CMTB93 44131470 Ki = 143 nM T21945 CYE20L 44131666 Ki = 663 nM T21945 CPR7L3 44133672 Ki = 140 nM T21945 CE3SD9 44133859 Ki = 25 nM T21945 CZ2VQ1 44133861 Ki = 413 nM T21945 C9P5XU 44133863 Ki = 921 nM T21945 C2G7AO 44134036 Ki = 27 nM T21945 C5YKI9 44134038 EC50 = 9 nM T21945 C6DQJ3 44134039 Ki = 181 nM T21945 C8RZX0 44134041 Ki = 1810 nM T21945 CW5Q9P 44143473 IC50 = 1930 nM T21945 CO0GC4 44157259 Ki > 6000 nM T21945 CGA8B4 44157339 Ki > 6000 nM T21945 C25DHI 44178203 Ki = 251.19 nM T21945 CI12UH 44188274 IC50 = 2 nM T21945 CT30BL 44188275 IC50 = 5850 nM T21945 CH7FJ6 44188689 Ki = 39.81 nM T21945 CSE8X3 44188690 Ki = 158.49 nM T21945 CY2Q9O 44188691 Ki = 31.62 nM T21945 C6FPM5 44188693 Ki = 79.43 nM T21945 CWR04I 44188695 Ki = 19.95 nM T21945 CJEG24 44188861 Ki = 199.53 nM T21945 C9XSI6 44189029 Ki = 316.23 nM T21945 C2AV1K 44190762 IC50 = 2160 nM T21945 C6WSI1 44204599 IC50 = 22.48 nM T21945 C2KJB0 44216880 Ki = 10 nM T21945 CA50PK 44219207 Ki = 1.585 nM T21945 CQY1J3 44219363 Ki = 158.49 nM T21945 CJX5T2 44219364 Ki = 398.11 nM T21945 C6SF0L 44219365 Ki = 25.12 nM T21945 CWP84D 44219367 Ki = 79.43 nM T21945 CVG5I0 44219517 Ki = 31.62 nM T21945 C1NQ2R 44219519 Ki = 31.62 nM T21945 CKMV39 44219520 Ki = 25.12 nM T21945 CA46YO 44230734 Ki = 11 nM T21945 CCK73R 44230855 IC50 = 8 nM T21945 CB5P7N 44230873 Ki = 8 nM T21945 CXI7Z8 44230875 Ki = 16 nM T21945 CU8MS7 44230877 Ki = 5 nM T21945 C67PRE 44231009 Ki = 1 nM T21945 C67WIP 44231010 Ki = 288 nM T21945 CCP13S 44231144 Ki = 5 nM T21945 CIBR82 44231149 Ki = 151 nM T21945 C8KE0I 44231252 IC50 = 7.4 nM T21945 CE12BT 44231265 Ki = 10 nM T21945 C0TF4H 44231266 Ki = 19 nM T21945 C7HCZ5 44231267 Ki = 71 nM T21945 CDZ8F4 44231268 Ki = 41 nM T21945 C0AW6X 44241240 IC50 = 7.7 nM T21945 C8AFN4 44241291 IC50 = 14 nM T21945 C63GVH 44241292 IC50 = 9.2 nM T21945 C9YZW2 44254588 IC50 = 18.6 nM T21945 C8OT6L 44254590 IC50 = 42.5 nM T21945 C6RO8P 44254675 IC50 = 39.4 nM T21945 C21AJO 44254678 IC50 = 91.9 nM T21945 C2R4VX 44254777 IC50 = 13.4 nM T21945 CR6KS9 44254860 IC50 = 7.8 nM T21945 C24WLR 44254964 IC50 = 17.5 nM T21945 C2EX8L 44255050 IC50 = 56 nM T21945 CG4T0O 44255052 IC50 = 66.7 nM T21945 C6HP5W 44255139 IC50 > 1000 nM T21945 CHD3K0 44267819 Ki = 3520 nM T21945 C8WZG7 44269522 Ki = 111 nM T21945 C0MCK3 44269548 Ki = 161 nM T21945 C96ZRI 44269549 Ki = 450 nM T21945 C5YE8A 44269598 Ki = 5.6 nM T21945 CI14GD 44269607 Ki = 2.5 nM T21945 CE20CZ 44275807 Ki = 9772.37 nM T21945 C2B8AN 44295896 IC50 = 0.8 nM T21945 CC3T9P 44295975 Ki = 22 nM T21945 CEO46F 44305466 Ki = 68 nM T21945 C97SYT 44305491 Ki = 640 nM T21945 CZG6F3 44305492 Ki = 208 nM T21945 CD3M2K 44307360 Ki = 1360 nM T21945 CUSR03 44307440 Ki = 118 nM T21945 C3WLT2 44307441 Ki > 20000 nM T21945 C7U8NC 44307585 Ki = 3024 nM T21945 C8RHD9 44308474 Ki = 330 nM T21945 C0LCV4 44308475 Ki = 2068 nM T21945 C0O2BH 44308682 IC50 = 266 nM T21945 CU0SQ8 44332340 IC50 = 620 nM T21945 C78AWT 44332801 IC50 = 296 nM T21945 CK68BR 44332802 IC50 = 109 nM T21945 CEG5D6 44332819 IC50 = 110 nM T21945 CICR35 44340153 Ki = 120 nM T21945 CJL61A 44340169 IC50 = 28 nM T21945 C40RKF 44340181 IC50 = 25 nM T21945 C78CFJ 44340203 IC50 = 34 nM T21945 CB34ZC 44340445 Ki = 68 nM T21945 CVWM21 44340483 Ki = 385 nM T21945 C4TSF5 44340484 Ki = 50 nM T21945 CQL94N 44340485 Ki = 316 nM T21945 C51NOI 44344091 Ki > 10000000 nM T21945 CX12US 44344115 Ki = 554000 nM T21945 C4PT6K 44344218 Ki = 235500 nM T21945 CX2O9B 44344235 Ki = 18400 nM T21945 CCI5T8 44354020 Ki > 10000 nM T21945 CGQ13N 44354021 Ki > 10000 nM T21945 C68QVH 44354105 IC50 = 173 nM T21945 C2TGL8 44354122 Ki > 10000 nM T21945 C4GVC5 44354236 IC50 = 1452 nM T21945 CFW7N2 44358674 IC50 = 7.3 nM T21945 CUN25S 44358675 IC50 = 16.3 nM T21945 C7BRY8 44358948 Ki = 20 nM T21945 CYI70C 44358978 Ki = 40 nM T21945 CYL37V 44358996 Ki = 36 nM T21945 CNU16S 44358997 Ki = 110 nM T21945 CWP87F 44359029 Ki = 70 nM T21945 C0HTE7 44359122 Ki = 67 nM T21945 CA1Q4M 44359155 Ki = 74 nM T21945 CS6O4C 44359156 Ki = 81 nM T21945 CDCU47 44359185 Ki = 78 nM T21945 CI0OX3 44359318 Ki = 160 nM T21945 CC2W7X 44359319 Ki = 42 nM T21945 CJ36NW 44364204 Ki = 55 nM T21945 C0O2NU 44364206 Ki = 86 nM T21945 CMA5D4 44364314 Ki = 460 nM T21945 C69BCI 44364358 Ki = 540 nM T21945 CL2M6Y 44364359 Ki = 170 nM T21945 C35MGZ 44364439 Ki = 4800 nM T21945 CLW8D9 44364455 Ki = 28 nM T21945 CRY94A 44370219 Ki > 10000 nM T21945 CWGQ58 44383909 Ki = 24 nM T21945 C24DSJ 44384117 Ki = 32 nM T21945 CX0V4W 44398372 Ki = 303 nM T21945 CA09EW 44404169 Ki > 200 nM T21945 C5Y8LB 44404175 Ki = 18 nM T21945 CM46ID 44404176 Ki = 79 nM T21945 CX02GP 44404182 Ki = 38 nM T21945 CV39CT 44404223 Ki = 11 nM T21945 C3KE9P 44404224 Ki = 150 nM T21945 CWD08P 44404228 Ki = 8 nM T21945 CG4P9S 44404235 Ki = 6 nM T21945 C4E6QN 44404238 Ki = 43 nM T21945 CVW0P1 44404239 Ki = 47 nM T21945 CZ9GU0 44404250 Ki = 44 nM T21945 CF8Z6A 44404254 Ki = 146 nM T21945 CN15FZ 44404255 Ki = 92 nM T21945 C30QXS 44404259 Ki = 21 nM T21945 C8U9NH 44404261 Ki = 150 nM T21945 CRSC86 44404262 Ki = 1430 nM T21945 CM7W1J 44404265 Ki = 9 nM T21945 CFP8D2 44404266 Ki > 200 nM T21945 C97CAH 44404269 Ki = 62 nM T21945 C5R7XB 44404273 Ki = 77 nM T21945 C5F2VA 44404274 Ki = 165 nM T21945 CGN87C 44404278 Ki > 200 nM T21945 CSO98W 44404279 Ki = 10 nM T21945 CRIG21 44404285 Ki = 7 nM T21945 CO57NJ 44404286 Ki = 17 nM T21945 CL6C2S 44404914 IC50 = 22 nM T21945 CSDN32 44405146 Ki = 627 nM T21945 C4DFS7 44405156 Ki = 308 nM T21945 CZI0A4 44405840 IC50 = 0.003 nM T21945 CR30FO 44405845 IC50 = 82700 nM T21945 C9TUH6 44405846 IC50 = 6430 nM T21945 CFT43Y 44405871 IC50 = 2020 nM T21945 CS2Q0A 44405875 IC50 = 23000 nM T21945 CR06US 44405876 IC50 = 3956 nM T21945 CG3WT6 44405893 IC50 = 62600 nM T21945 CDF9N4 44405897 IC50 = 66300 nM T21945 C4GN3T 44405898 IC50 = 41500 nM T21945 CA3I0W 44407714 Ki > 10000 nM T21945 CIH46L 44408412 IC50 > 100 nM T21945 CK6O7A 44408415 IC50 > 100 nM T21945 CV3QD5 44408434 IC50 > 100 nM T21945 C7T6WF 44408435 IC50 > 100 nM T21945 CJ3NS2 44408441 IC50 > 100 nM T21945 CT52PU 44408442 IC50 > 100 nM T21945 CDQ34O 44408477 IC50 > 100 nM T21945 CI3Z8X 44408529 IC50 > 100 nM T21945 CYP8A5 44408580 IC50 > 100 nM T21945 CA3P6K 44408581 IC50 > 100 nM T21945 C6F5EC 44408582 IC50 > 100 nM T21945 CKX2P8 44408664 IC50 = 650 nM T21945 C3C9PW 44408718 IC50 = 3200 nM T21945 CK9U7V 44408719 IC50 = 2900 nM T21945 C83DCF 44408748 IC50 = 2100 nM T21945 CQ64UC 44408749 IC50 = 1800 nM T21945 C14BYG 44408753 IC50 = 920 nM T21945 CI0JZ2 44408756 IC50 = 60 nM T21945 C9U3TR 44408757 IC50 = 960 nM T21945 C6LTD5 44408760 IC50 = 760 nM T21945 CYAC79 44408761 IC50 = 680 nM T21945 CX2S0E 44408762 IC50 = 980 nM T21945 C3QCP2 44408802 IC50 = 4200 nM T21945 CLJ3U7 44408856 IC50 = 1100 nM T21945 C5K8NB 44408857 IC50 = 5000 nM T21945 C2QMD8 44408858 IC50 = 11500 nM T21945 CI3ZS8 44408859 IC50 = 20300 nM T21945 C1ZPY7 44408870 IC50 = 1150 nM T21945 C8ZH4C 44408871 IC50 = 1500 nM T21945 C2J1KW 44408875 IC50 = 2000 nM T21945 CZ8G2B 44408876 IC50 = 2100 nM T21945 CKR78J 44408885 IC50 = 2100 nM T21945 CC9D8S 44408886 IC50 = 9100 nM T21945 CW7VA3 44408917 IC50 = 1250 nM T21945 CBS73M 44408918 IC50 = 880 nM T21945 CQ45GH 44408921 IC50 = 9600 nM T21945 CKM7O2 44408922 IC50 = 450 nM T21945 C13IEG 44408925 IC50 = 310 nM T21945 CE5AC6 44408926 IC50 = 310 nM T21945 C2D5WU 44408969 IC50 = 11 nM T21945 CG87PW 44409290 Ki > 1000 nM T21945 C1GHS5 44410092 Ki = 30 nM T21945 C6MKX5 44410093 Ki = 11.9 nM T21945 C6AS4M 44410096 Ki = 5.2 nM T21945 CG48JW 44410236 Ki = 7.7 nM T21945 CXK2S9 44410237 Ki = 54.4 nM T21945 CFEN06 44410241 Ki = 3.7 nM T21945 C24AHO 44411099 Ki = 690 nM T21945 C2EQ1I 44411140 Ki = 3.3 nM T21945 CCBK16 44411148 Ki = 150 nM T21945 C7D8MV 44411168 Ki = 86 nM T21945 CDH1U9 44411170 Ki = 4.1 nM T21945 C5Z3ES 44411177 Ki = 6.1 nM T21945 CQA1W4 44411179 Ki = 43 nM T21945 C60ECT 44411185 Ki = 78 nM T21945 CY0U6V 44411206 Ki = 190 nM T21945 CI6B1W 44411208 Ki = 4.8 nM T21945 C1VHP7 44411215 Ki = 15 nM T21945 C9GW7B 44411217 Ki = 6 nM T21945 C1R3LU 44411219 Ki = 42.1 nM T21945 C3M7RB 44411224 Ki = 2 nM T21945 C0J6WV 44411226 Ki = 420 nM T21945 CT7D0B 44411228 Ki = 1.8 nM T21945 C7TH4P 44411230 Ki = 5.4 nM T21945 C5FYQ9 44411235 Ki = 5.5 nM T21945 CI8MC6 44411239 Ki = 9.6 nM T21945 CFUV50 44411241 Ki = 9.7 nM T21945 CUFD63 44411249 Ki = 13.3 nM T21945 C9BV1K 44411254 Ki = 15.9 nM T21945 CM6RO7 44411258 Ki = 8.3 nM T21945 CE5A4F 44411296 Ki = 2.7 nM T21945 CR3P8E 44411314 Ki = 9.8 nM T21945 C8GD7M 44411395 Ki = 1.4 nM T21945 C42XFV 44411397 Ki = 3.3 nM T21945 CHU4D8 44411449 Ki = 255 nM T21945 CTO82V 44411451 Ki = 300 nM T21945 CWN14V 44411456 Ki = 5.1 nM T21945 CIG3V6 44411460 Ki = 3.1 nM T21945 CW3KE8 44411466 Ki = 6 nM T21945 CTQ19K 44411482 Ki = 42 nM T21945 C5ZN4X 44411491 Ki = 20 nM T21945 CV2S7W 44411499 Ki = 175 nM T21945 C6CW9U 44411501 Ki = 2.2 nM T21945 CC5Z7V 44411505 Ki = 7.1 nM T21945 C6OS1M 44411507 Ki = 145 nM T21945 CH8W2F 44411510 Ki = 3.6 nM T21945 CF4O1I 44411514 Ki = 3.4 nM T21945 C21MSX 44411516 Ki = 1060 nM T21945 C4DZ1I 44411518 Ki = 61 nM T21945 CW0DM3 44411520 Ki = 6.5 nM T21945 C9JXM6 44411522 Ki = 6.2 nM T21945 C0DHC7 44411524 Ki = 95.9 nM T21945 CU8M4K 44411526 Ki = 8.3 nM T21945 C8XF4A 44411527 Ki = 6.1 nM T21945 C6PR1D 44411536 Ki = 4.2 nM T21945 C2GV3H 44411541 Ki = 51 nM T21945 CIBG87 44413825 Ki > 2000 nM T21945 CFN48L 44413826 Ki = 1400 nM T21945 CA97VC 44413836 Ki = 1160 nM T21945 CLG5H8 44413837 Ki > 2000 nM T21945 CCY43Q 44413856 Ki = 710 nM T21945 CW0VE9 44413857 Ki = 500 nM T21945 C05UKL 44413866 Ki = 490 nM T21945 CCJ4X1 44413903 Ki > 2000 nM T21945 C81IAE 44413904 Ki = 1060 nM T21945 C5Z2GC 44413925 Ki > 2000 nM T21945 C3BMI9 44413953 Ki > 2000 nM T21945 C18JHP 44413959 Ki = 1520 nM T21945 C3IE4V 44414667 IC50 > 400 nM T21945 CQ3C7F 44414684 IC50 = 270 nM T21945 CNR87Z 44414690 IC50 = 25 nM T21945 CCL7Y9 44414691 IC50 = 22 nM T21945 CM9V8F 44414692 IC50 = 94 nM T21945 CQD2S5 44414696 IC50 = 38 nM T21945 CM6D5P 44414704 IC50 = 28 nM T21945 CZ9LM3 44414707 IC50 = 31 nM T21945 CE85AH 44414731 IC50 = 340 nM T21945 C2BYE0 44414733 IC50 > 400 nM T21945 C9XIR1 44414734 IC50 = 61 nM T21945 C9FCZ2 44414748 IC50 = 120 nM T21945 C8RN6K 44414749 IC50 = 21 nM T21945 C81QHB 44414760 IC50 > 400 nM T21945 CV37KC 44414761 IC50 = 120 nM T21945 CUK97V 44414762 IC50 = 130 nM T21945 CI8NH6 44414763 IC50 = 38 nM T21945 C3LJ7N 44414780 IC50 = 82 nM T21945 CY5Q9A 44414800 IC50 = 75 nM T21945 C3RZ0N 44414809 IC50 = 15 nM T21945 CPR9Y5 44414810 IC50 = 45 nM T21945 CF8Q6Y 44414836 IC50 = 19 nM T21945 CWZ3E4 44414859 IC50 = 76 nM T21945 CA58NQ 44414873 IC50 = 8.8 nM T21945 CHCQ59 44414875 IC50 = 100 nM T21945 CVTQ68 44416033 Ki = 2.94 nM T21945 CZ6WJ8 44416034 Ki = 4.84 nM T21945 CRA8M1 44416084 Ki = 5.87 nM T21945 C1BF0K 44416103 Ki = 25.5 nM T21945 C9Q5UZ 44416104 Ki = 12.53 nM T21945 C9UDS3 44416105 Ki = 13.03 nM T21945 CHF6L7 44417598 Ki = 102.2 nM T21945 CK5PZ8 44417599 Ki = 31.7 nM T21945 CRZK78 44418862 Ki = 14 nM T21945 CXA51W 44419295 Ki = 1390 nM T21945 CLA67J 44419296 Ki = 497 nM T21945 C82VQX 44419298 Ki = 381 nM T21945 CRAK93 44419299 Ki = 5007 nM T21945 CZT81O 44419300 Ki = 317 nM T21945 C2WDJ5 44419301 Ki = 524 nM T21945 C85OTF 44419303 Ki = 1052 nM T21945 CZ5O8Y 44419306 Ki = 1379 nM T21945 CXP1A6 44419308 Ki = 9261 nM T21945 CM3K1F 44419314 Ki = 37 nM T21945 CG8F3J 44419327 Ki = 39 nM T21945 CJR7P1 44419328 Ki = 233 nM T21945 C7DQL6 44419331 Ki = 95 nM T21945 CVMF25 44419335 Ki = 3449 nM T21945 C59ZPV 44419340 Ki = 1230 nM T21945 C71CPW 44419344 Ki = 1480 nM T21945 CM1WZ9 44419345 Ki = 876 nM T21945 CJHN07 44421413 Ki = 271 nM T21945 CEHO31 44421414 Ki = 741 nM T21945 C2WE3K 44421423 Ki = 16.2 nM T21945 C1S3RH 44421438 Ki = 280 nM T21945 CSIN57 44421439 Ki = 1930 nM T21945 CQI4V3 44421455 Ki = 160 nM T21945 C2BEZ9 44421482 Ki = 7800 nM T21945 C7PCA5 44421483 Ki = 191 nM T21945 CNYK42 44421484 Ki = 6000 nM T21945 CB17LT 44421485 Ki = 46000 nM T21945 CE6G3H 44421486 Ki = 61 nM T21945 CL6M9V 44421497 Ki = 280 nM T21945 CSU23Q 44421500 Ki = 3700 nM T21945 CCGM26 44422453 Ki = 8.29 nM T21945 CV43NH 44427225 IC50 = 2000 nM T21945 CGX49R 44427889 Ki = 28 nM T21945 C7I2MZ 44427901 Ki = 28 nM T21945 CGOD89 44429174 Ki = 3910 nM T21945 C6BW5V 44429184 Ki = 2300 nM T21945 CIJ5R2 44429185 Ki = 2500 nM T21945 C6OVA2 44429187 Ki = 10000 nM T21945 CNP37Y 44429189 Ki = 11000 nM T21945 C8SR0G 44429190 Ki = 178000 nM T21945 C53AFL 44429191 Ki = 285000 nM T21945 CN4UT8 44429192 Ki = 26000 nM T21945 C5HK8Y 44429193 Ki = 550000 nM T21945 C7J6GA 44429194 Ki = 789000 nM T21945 CK9H1C 44429195 Ki = 2884000 nM T21945 CQA0W7 44429197 Ki = 240000 nM T21945 CV9M4N 44429198 Ki = 247000 nM T21945 CUH0B6 44429199 Ki = 111000 nM T21945 CS2ER7 44429200 Ki = 4900 nM T21945 CE2M3T 44429201 Ki = 314000 nM T21945 CE31CZ 44429202 Ki = 339000 nM T21945 CF5CO6 44429203 Ki = 10000 nM T21945 CJ9VZ1 44429204 Ki = 215000 nM T21945 CJ5F4X 44429205 Ki = 1100000 nM T21945 CLK84J 44429206 Ki = 2540000 nM T21945 CH50DU 44429207 Ki = 2500000 nM T21945 C1Z7KB 44429209 Ki = 2110000 nM T21945 C7OQT6 44429210 Ki = 2020000 nM T21945 CI46CX 44429212 Ki = 499000 nM T21945 CA2HN0 44429214 Ki = 121000 nM T21945 CE30YG 44429218 Ki = 4720 nM T21945 CM5HG8 44429219 Ki = 20000 nM T21945 C4I1GO 44429221 Ki = 85000 nM T21945 CDGP34 44429222 Ki = 68000 nM T21945 CW7L3V 44429226 Ki = 3900 nM T21945 CKF60U 44429227 Ki = 255000 nM T21945 CX4EM1 44429392 Ki = 658000 nM T21945 C3JNX9 44429393 Ki = 675000 nM T21945 CH9W4Z 44429395 Ki = 719000 nM T21945 C3O9DN 44429396 Ki = 1360000 nM T21945 CO29HT 44429397 Ki = 991000 nM T21945 C75HYO 44429399 Ki = 439000 nM T21945 C7TXV4 44429400 Ki = 51000 nM T21945 CBR73H 44429401 Ki = 94000 nM T21945 CG9N0T 44429402 Ki = 62000 nM T21945 CQG41A 44430844 IC50 = 49 nM T21945 CF4BK0 44430849 IC50 = 37 nM T21945 C82VMO 44430851 IC50 = 390 nM T21945 C6CD3M 44431728 Ki = 1.78 nM T21945 CT2UJ0 44431732 Ki = 4.88 nM T21945 CE2QP4 44431734 Ki = 1.98 nM T21945 CHR6F7 44431736 Ki = 4.67 nM T21945 CH6B3Y 44431739 Ki = 1.86 nM T21945 CF42IC 44434165 Ki = 250 nM T21945 C50ZDW 44439863 Ki = 121 nM T21945 CZ9F1A 44440497 Ki = 1245 nM T21945 CF8K5H 44441067 Ki = 460 nM T21945 C6P8RJ 44441332 IC50 = 15 nM T21945 CDEY23 44441334 IC50 = 9 nM T21945 COBN96 44441335 IC50 = 5 nM T21945 C23BGW 44441336 IC50 = 3 nM T21945 C92ABN 44441338 IC50 = 8 nM T21945 C6K8ZB 44441339 IC50 = 12 nM T21945 CJ2S0W 44441340 IC50 = 144 nM T21945 C1R0DN 44441341 IC50 = 7 nM T21945 C9FB6Y 44441345 IC50 = 4 nM T21945 CZ34LI 44441346 IC50 = 5 nM T21945 C2GAV7 44441348 IC50 = 20 nM T21945 CWH92R 44441349 IC50 = 11 nM T21945 C61VKY 44441350 IC50 = 13 nM T21945 CF4A8D 44441351 IC50 = 7 nM T21945 CD30KT 44441353 IC50 = 40 nM T21945 C8ZJU5 44443873 Ki = 300000 nM T21945 C4X5GY 44443875 Ki = 410000 nM T21945 CI0Q6D 44443877 Ki = 210000 nM T21945 COC4G7 44443878 Ki = 50000 nM T21945 C9JB8C 44443887 Ki = 8000 nM T21945 C3Q8RJ 44443888 Ki = 250000 nM T21945 CCP50E 44443889 Ki = 9200 nM T21945 CSF8J3 44443890 Ki = 18000 nM T21945 CRB6J3 44443891 Ki = 12000 nM T21945 C0EI1N 44443892 Ki = 130000 nM T21945 CZUT06 44443893 Ki = 26000 nM T21945 CWB8E6 44443894 Ki = 9000 nM T21945 CDW62E 44443895 Ki = 5800 nM T21945 CR1AP8 44443896 Ki = 170000 nM T21945 CVK42D 44443897 Ki = 85000 nM T21945 CEI6Y9 44443898 Ki = 33000 nM T21945 C2WC8G 44443899 Ki = 42000 nM T21945 C03MYS 44443900 Ki = 61000 nM T21945 C6FY0T 44444517 IC50 = 68000 nM T21945 CMEO07 44444525 IC50 = 19000 nM T21945 C92VUT 44444530 IC50 = 39000 nM T21945 CG0TP9 44444534 IC50 = 8700 nM T21945 CCMZ42 44444540 IC50 = 560 nM T21945 C0YOW4 44448355 IC50 = 12 nM T21945 CZS5L9 44448356 IC50 = 200 nM T21945 CG4D7J 44448357 IC50 = 8.3 nM T21945 C9RJX0 44448358 IC50 = 37 nM T21945 C7AW4C 44448387 IC50 = 8.2 nM T21945 C15HXQ 44448388 IC50 = 44 nM T21945 C1OQ2Y 44448389 IC50 = 3.9 nM T21945 CE80KR 44448391 IC50 = 64 nM T21945 CQV39U 44448392 IC50 = 110 nM T21945 CPV4Z3 44448423 IC50 = 1100 nM T21945 CFC8I2 44448425 IC50 = 2.8 nM T21945 CM8QA0 44448426 IC50 = 20 nM T21945 C1LIQ2 44448427 IC50 = 2.7 nM T21945 CW51IM 44448465 IC50 = 5.6 nM T21945 C1MIQ3 44448466 IC50 = 100 nM T21945 CO4GZ7 44448467 IC50 > 10000 nM T21945 COE35W 44448468 IC50 = 170 nM T21945 C5GTQ1 44448470 IC50 = 3700 nM T21945 CJ8X7A 44448508 IC50 = 2200 nM T21945 CKO0F9 44448509 IC50 = 150 nM T21945 C36MOD 44448511 IC50 = 1500 nM T21945 CCR7Q2 44448512 IC50 = 65 nM T21945 CPS91V 44448544 IC50 = 560 nM T21945 CO9U4F 44448545 IC50 = 270 nM T21945 CM6W2E 44448546 IC50 = 1500 nM T21945 CWA0E4 44448547 IC50 = 29 nM T21945 C9HVB8 44448548 IC50 = 40 nM T21945 CSYB74 44448582 IC50 = 76 nM T21945 CF0ZG2 44448584 IC50 = 2.9 nM T21945 C67GMI 44449234 IC50 = 38 nM T21945 C3RMF8 44449236 IC50 = 26 nM T21945 CM4F7Z 44449237 IC50 = 85 nM T21945 C2UQI1 44449238 IC50 = 26 nM T21945 C3HS9U 44449239 IC50 = 51 nM T21945 CQN4Z9 44449267 IC50 = 36 nM T21945 CZ3UA5 44449268 Ki = 22 nM T21945 C8FBZ0 44449269 IC50 = 246 nM T21945 CS6R9X 44449270 IC50 = 22 nM T21945 CKH31F 44449272 IC50 = 18 nM T21945 CD4J9E 44449296 IC50 = 86 nM T21945 CGK7O1 44449297 IC50 = 47 nM T21945 CVZ39S 44449298 IC50 = 83 nM T21945 C2O9KI 44449307 IC50 = 4.5 nM T21945 C9MU1V 44449332 IC50 = 282 nM T21945 CJC38Z 44449333 IC50 = 32 nM T21945 C6X4JZ 44449340 IC50 = 18 nM T21945 CCB54W 44449341 IC50 = 21 nM T21945 C1CPD4 44449368 IC50 = 3.5 nM T21945 CR4OB8 44449369 IC50 = 47 nM T21945 C7W4XU 44449370 IC50 = 160 nM T21945 CC2ZK5 44449371 IC50 = 4 nM T21945 CZSE46 44449372 IC50 = 73 nM T21945 CZY4G7 44449373 IC50 = 47 nM T21945 CH48QG 44449395 IC50 = 8.1 nM T21945 C2YG0E 44449396 IC50 = 3.2 nM T21945 CD9LA2 44449397 IC50 = 4.4 nM T21945 CWG79A 44449398 IC50 = 3.9 nM T21945 CW98KH 44449399 IC50 > 10000 nM T21945 CYM7I3 44449400 IC50 > 10000 nM T21945 CK9UP5 44449401 IC50 > 10000 nM T21945 C8EJ1M 44449434 IC50 = 5.9 nM T21945 C6KR7N 44449435 IC50 = 6400 nM T21945 C59NSQ 44449436 IC50 > 10000 nM T21945 C2QF0K 44449437 IC50 > 10000 nM T21945 C2Z6IM 44449438 IC50 > 10000 nM T21945 CJL4G7 44449462 IC50 = 7.1 nM T21945 C50SKP 44449464 IC50 = 14 nM T21945 CT76PB 44449465 IC50 = 4.4 nM T21945 COU68C 44449519 IC50 = 5.2 nM T21945 C0X2RW 44449521 IC50 = 2.9 nM T21945 CG2AD9 44449552 IC50 = 6.3 nM T21945 CY0B5K 44449554 IC50 = 20 nM T21945 CHA59Q 44449589 IC50 = 4.2 nM T21945 CDQ89E 44449590 IC50 = 15 nM T21945 C53EYA 44449619 IC50 = 7 nM T21945 CUXK25 44449620 IC50 = 7.6 nM T21945 C7KZ5C 44449623 IC50 = 160 nM T21945 CZ1L4G 44449624 IC50 = 12 nM T21945 C8K3XF 44449625 IC50 = 7.1 nM T21945 CYRM03 44449651 IC50 = 40 nM T21945 C15DIZ 44449652 IC50 = 80 nM T21945 CWO0H5 44449656 IC50 = 17 nM T21945 C7ENK5 44449717 IC50 = 159 nM T21945 C41WXJ 44449718 IC50 = 25 nM T21945 C7KQ4B 44449719 IC50 = 394 nM T21945 CC5K0E 44449720 IC50 = 257 nM T21945 C2KA8J 44449721 IC50 > 400 nM T21945 C2QP0Z 44449729 IC50 = 14 nM T21945 C3VE2D 44449768 Ki = 610 nM T21945 C3FP2I 44449792 Ki = 6 nM T21945 C83ICG 44449794 Ki = 420 nM T21945 CS9ZO8 44449911 Ki = 15 nM T21945 C50ZLO 44449944 Ki = 275 nM T21945 CJ83BL 44450087 Ki = 16 nM T21945 CW9P8L 44450088 Ki = 180 nM T21945 CB8W3Q 44450089 Ki = 29 nM T21945 C26WAJ 44450090 Ki = 84 nM T21945 CMKF97 44450118 Ki = 22 nM T21945 C35FRM 44450119 Ki = 9 nM T21945 CK1B8X 44450120 Ki = 160 nM T21945 C4AUT7 44450121 Ki = 28 nM T21945 CJOI42 44450152 Ki = 210 nM T21945 C6FBZ1 44450153 Ki = 12 nM T21945 C52HPA 44450154 Ki = 350 nM T21945 C9SB0X 44450155 Ki = 17 nM T21945 CAW6S7 44450181 Ki = 130 nM T21945 CJ8KS4 44450182 Ki = 12 nM T21945 C4M0PG 44450184 Ki = 860 nM T21945 C4KE7B 44450185 Ki = 10 nM T21945 C4VL3W 44450211 Ki = 12 nM T21945 CSQR06 44450212 Ki = 830 nM T21945 CXR4G1 44450213 Ki = 18 nM T21945 CTX1Q7 44452747 Ki = 296 nM T21945 CIS3J5 44452748 Ki = 461 nM T21945 COAL13 44452772 Ki = 921 nM T21945 C42KFD 44452774 Ki = 366 nM T21945 CGR0B6 44452775 Ki = 27 nM T21945 C80CWR 44452935 Ki = 10 nM T21945 CY01KA 44452990 Ki = 159 nM T21945 C8Q7OP 44452992 Ki = 438 nM T21945 CV92RP 44452994 Ki = 13 nM T21945 CLSI34 44453016 Ki = 131 nM T21945 CKZN93 44453017 Ki = 82 nM T21945 CB1OY5 44453042 Ki = 255 nM T21945 C2HFJ7 44453043 Ki = 58 nM T21945 CY38AM 44453067 Ki = 232 nM T21945 CBP25X 44453068 Ki = 194 nM T21945 CR4F7O 44453093 Ki = 951 nM T21945 C01QKJ 44453119 Ki = 179 nM T21945 CB06JG 44454485 IC50 = 4900 nM T21945 CISA76 44454488 IC50 = 8000 nM T21945 CE1X7O 44454489 IC50 = 6100 nM T21945 CYRU93 44454493 IC50 = 860 nM T21945 CKJ2D3 44454526 IC50 = 360 nM T21945 CB9M0F 44454528 IC50 = 41 nM T21945 CYCB65 44454556 IC50 > 10000 nM T21945 CH4JN9 44454557 IC50 = 1400 nM T21945 CJB41D 44454559 IC50 = 570 nM T21945 CQ87FZ 44454585 IC50 > 10000 nM T21945 C8LR9P 44454660 IC50 = 150 nM T21945 C3T5HK 44454663 IC50 = 12 nM T21945 C89SJY 44454690 IC50 > 10000 nM T21945 CYZ39A 44454694 IC50 > 10000 nM T21945 C0QVN8 44454719 IC50 > 10000 nM T21945 C01XOI 44454744 IC50 = 8.4 nM T21945 C1H0FI 44454746 IC50 = 8100 nM T21945 C43QBZ 44454747 IC50 = 2600 nM T21945 CEY3T6 44454767 IC50 = 21 nM T21945 C8FBC2 44454794 IC50 > 10000 nM T21945 CJBD47 44454795 IC50 = 130 nM T21945 C4WOL9 44454797 IC50 = 2900 nM T21945 CU49TR 44454860 IC50 = 2300 nM T21945 COX3W0 44454862 IC50 = 170 nM T21945 CQF13W 44454863 IC50 = 960 nM T21945 CU21QR 44454893 IC50 = 63 nM T21945 CU8K7O 44454894 IC50 = 200 nM T21945 CVU57D 44454896 IC50 = 8400 nM T21945 C1P5VQ 44454931 IC50 = 180 nM T21945 CZ2X0T 44454932 IC50 > 10000 nM T21945 CXC09Y 44454967 IC50 > 10000 nM T21945 C75SEP 44454968 IC50 = 6248 nM T21945 C5LN9M 44454971 IC50 = 3776 nM T21945 CIH52C 44455025 IC50 = 3776 nM T21945 CI5T8S 44455135 IC50 = 3789 nM T21945 CGI6A7 44455136 IC50 = 1565 nM T21945 CM9OW7 44455170 IC50 = 8999 nM T21945 C8E4AF 44455171 IC50 = 898 nM T21945 CH4N8R 44455206 IC50 > 10000 nM T21945 CEZR53 44455270 IC50 = 3873 nM T21945 CVDA26 44455301 IC50 = 3861 nM T21945 C0UC6P 44455338 IC50 = 5948 nM T21945 C89COF 44455373 IC50 > 10000 nM T21945 CRFJ58 44455391 IC50 = 4495 nM T21945 CMNX58 44455445 IC50 > 10000 nM T21945 CC09EJ 44455512 Ki = 112 nM T21945 C6YQU9 44455589 IC50 = 11 nM T21945 C9PG3H 44455590 IC50 = 25 nM T21945 C1BR2G 44455619 IC50 = 26 nM T21945 CO1X6Z 44455620 IC50 = 17 nM T21945 C8F5CI 44455622 IC50 = 46 nM T21945 C0EM9R 44455651 IC50 = 17 nM T21945 CW7E6X 44455652 IC50 = 33 nM T21945 C3W1EZ 44455653 IC50 > 400 nM T21945 CI4K0E 44455654 IC50 = 84 nM T21945 CZV45C 44455655 IC50 = 38 nM T21945 C0L9YB 44455677 IC50 = 62 nM T21945 CV10IJ 44455678 IC50 = 78 nM T21945 CK47LB 44455681 IC50 > 400 nM T21945 CIW6A1 44455707 IC50 = 429 nM T21945 CR24HA 44455708 IC50 = 157 nM T21945 CJM9O8 44455710 IC50 = 300 nM T21945 COV02B 44455738 IC50 = 46 nM T21945 C3CXW8 44455739 IC50 = 14 nM T21945 CO4B1F 44455740 IC50 = 78 nM T21945 C3I6TO 44455742 IC50 = 21 nM T21945 C76JRV 44455761 IC50 = 50 nM T21945 CSX82U 44455763 IC50 = 15 nM T21945 C16SFL 44455822 Ki = 420 nM T21945 C08MBY 44456312 Ki = 82 nM T21945 CS74YL 44457050 Ki = 1.35 nM T21945 C36OQY 44457051 Ki = 1 nM T21945 CKI8L5 44457058 Ki = 1.32 nM T21945 CQS23B 44457059 Ki = 2.06 nM T21945 CC9ZF1 44462051 Ki = 1.4 nM T21945 CN3H5R 44462082 Ki = 36 nM T21945 CL9O8M 44462783 IC50 = 6 nM T21945 C91PCM 44466344 Ki = 10 nM T21945 CZA36I 44466345 Ki = 79.43 nM T21945 C63XKS 44467026 Ki = 3.981 nM T21945 CH4WM3 44467027 Ki = 12.59 nM T21945 C3T4BX 44467028 Ki = 12.59 nM T21945 CG4R7A 44467101 Ki = 251.19 nM T21945 CW2K9E 44467103 Ki = 6.31 nM T21945 CL0JR9 44467104 Ki = 1000 nM T21945 C4CX9E 44467173 Ki = 1584.89 nM T21945 CG4H1R 44467174 Ki = 39.81 nM T21945 CLU6A0 44467177 Ki = 25.12 nM T21945 C4RBV8 44467889 Ki = 15.85 nM T21945 CJB37C 44467892 Ki = 50.12 nM T21945 CF4ZM8 44467957 Ki = 7.943 nM T21945 CTO9R8 44467960 Ki = 199.53 nM T21945 CM5OT7 44473055 Ki = 9 nM T21945 CR74ZI 44473056 Ki = 208 nM T21945 C6PT2I 44473057 IC50 = 1092 nM T21945 C7CEY4 44473058 Ki = 21 nM T21945 CRZK08 44473059 IC50 = 12 nM T21945 CV3TN8 44473060 IC50 = 707 nM T21945 CM6Q7W 44474580 Ki = 75.7 nM T21945 C73XSD 44474582 Ki = 27.8 nM T21945 C68VDK 44474583 Ki = 153 nM T21945 C21WPR 44474586 Ki = 1.19 nM T21945 C3DHG0 44511399 IC50 = 69 nM T21945 CU9MO1 44539110 Ki = 0.1259 nM T21945 CAL8V3 44539203 Ki = 79.43 nM T21945 CO1E5C 44539964 IC50 = 13.3 nM T21945 CLMY52 44539967 IC50 = 19.8 nM T21945 CLO73R 44540428 IC50 = 264 nM T21945 CV92IJ 44541354 IC50 = 16 nM T21945 C5Q3NI 44542504 IC50 > 100 nM T21945 C5F1UC 44542505 Ki > 10000 nM T21945 CYX7H5 44542510 IC50 = 900 nM T21945 C71QGD 44542511 Ki > 10000 nM T21945 C8V7UL 44542657 IC50 = 360 nM T21945 C6ECJ1 44542658 IC50 = 86 nM T21945 C2EDU6 44542955 IC50 > 100 nM T21945 CTW5I9 44542956 Ki > 10000 nM T21945 C03MXJ 44543264 IC50 = 6480 nM T21945 CL5UK7 44543265 Ki = 4600 nM T21945 CBL30Z 44543269 Ki = 3800 nM T21945 CHIY92 44543270 Ki > 10000 nM T21945 C94MOI 44559129 IC50 = 30000 nM T21945 C1YIC9 44560434 Ki = 553 nM T21945 C7G9WM 44560436 Ki = 552 nM T21945 C35XEU 44560438 Ki > 2000 nM T21945 CBTX17 44560440 Ki > 2000 nM T21945 CB0K6T 44560442 Ki = 466 nM T21945 CWCT08 44560444 Ki = 349 nM T21945 C69ETG 44560446 Ki = 788 nM T21945 CK2PD5 44560493 Ki = 1030 nM T21945 C2SZ1B 44560495 Ki > 2000 nM T21945 C9U5SE 44560498 Ki = 455 nM T21945 CNK4F6 44560500 Ki = 519 nM T21945 CU05HZ 44560502 Ki > 2000 nM T21945 C87VZD 44560504 Ki > 2000 nM T21945 CV0BF4 44560506 Ki > 2000 nM T21945 CS9N0U 44560575 IC50 = 4000 nM T21945 CYNS29 44560577 IC50 = 2000 nM T21945 CF5BX9 44560599 Ki = 1300 nM T21945 CNF81T 44560602 Ki = 435 nM T21945 CWB6S3 44560604 Ki = 454 nM T21945 CJQ4R5 44560606 Ki = 677 nM T21945 C7TO9F 44560608 Ki = 840 nM T21945 C17ZEN 44560622 IC50 = 800 nM T21945 CN1K6R 44560623 IC50 = 4000 nM T21945 C9BV0O 44560624 IC50 = 1600 nM T21945 CY72NM 44560625 IC50 = 6000 nM T21945 C0FW5J 44560626 IC50 = 660 nM T21945 CLW2R6 44560627 IC50 = 150 nM T21945 CI1XD4 44560628 IC50 = 3000 nM T21945 C1NCT4 44560653 Ki = 1100 nM T21945 C8MPN0 44560655 Ki = 770 nM T21945 CWG57V 44560657 Ki = 347 nM T21945 CH79ZT 44560659 Ki = 357 nM T21945 C51DKQ 44560671 IC50 = 3000 nM T21945 CBMT59 44560672 IC50 = 2000 nM T21945 C1R8PQ 44560673 IC50 = 1100 nM T21945 CGK29S 44560675 IC50 = 72 nM T21945 CG4YN5 44560676 IC50 = 150 nM T21945 CNM1Q6 44560708 IC50 = 430 nM T21945 CG6FL1 44560709 IC50 = 200 nM T21945 CL9J2E 44560710 IC50 = 190 nM T21945 C36IOW 44560711 IC50 = 160 nM T21945 CLM2F8 44560712 IC50 = 630 nM T21945 C3OG8F 44560713 IC50 = 520 nM T21945 C9B5CE 44560714 IC50 = 950 nM T21945 CP7RQ8 44562623 IC50 = 75 nM T21945 CHE68Z 44562624 IC50 = 77 nM T21945 CR4TG7 44562625 IC50 = 11 nM T21945 CH32FI 44562626 IC50 = 5 nM T21945 CX1P3L 44562627 IC50 = 17 nM T21945 C0S8ZG 44562682 IC50 = 2 nM T21945 C2HKE0 44562772 IC50 = 300 nM T21945 C50WKO 44562773 IC50 = 3 nM T21945 C3JD7Y 44562774 IC50 = 2 nM T21945 CS0LD7 44562775 IC50 = 3 nM T21945 C7AC8Z 44562776 IC50 = 5 nM T21945 CU6G4W 44562777 IC50 = 7 nM T21945 CCA0H2 44562815 IC50 = 5 nM T21945 CQ0I5R 44562816 IC50 = 4 nM T21945 CC1IF3 44562817 IC50 = 4 nM T21945 CR28PD 44563213 IC50 = 3 nM T21945 CU4PD5 44563214 IC50 = 3 nM T21945 CGKL94 44563257 IC50 = 10 nM T21945 C8TYL3 44563258 IC50 = 30 nM T21945 C8XUD6 44563259 IC50 > 10000 nM T21945 CIG6Z4 44563260 IC50 = 700 nM T21945 C9VFW6 44563261 IC50 = 2800 nM T21945 C9N0RT 44563646 Ki = 109.9 nM T21945 CEG7S1 44563647 Ki = 101.3 nM T21945 C41KWG 44563667 Ki = 67.5 nM T21945 CI6A1Q 44563668 Ki = 30.2 nM T21945 CL83PU 44563669 Ki = 1180 nM T21945 CJD73U 44565305 IC50 = 7441 nM T21945 CM8LR1 44568174 IC50 > 10000 nM T21945 CCRI61 44568175 IC50 = 680 nM T21945 CB3VF8 44568176 IC50 = 1500 nM T21945 C6T2BK 44568293 IC50 = 1400 nM T21945 CA1NJ9 44568294 IC50 = 2700 nM T21945 CA21KI 44568295 IC50 = 4900 nM T21945 CX50DP 44568296 IC50 = 50 nM T21945 COB14G 44568297 IC50 = 430 nM T21945 C3I6FM 44568320 IC50 = 130 nM T21945 C4QYH2 44568321 IC50 = 1050 nM T21945 CKT30F 44568322 IC50 > 10000 nM T21945 C1HA7U 44568323 IC50 = 3000 nM T21945 C9CJP2 44568324 IC50 > 10000 nM T21945 C81XJM 44568325 IC50 = 6400 nM T21945 C3SW7N 44568349 IC50 = 2000 nM T21945 CLTG36 44568350 IC50 = 530 nM T21945 C9MNC0 44568351 IC50 = 70 nM T21945 CB58VS 44568378 IC50 = 2900 nM T21945 CYN68I 44568379 IC50 = 510 nM T21945 CY3NQ8 44568652 IC50 = 200 nM T21945 C02GHU 44568653 IC50 = 1300 nM T21945 C8HNK7 44568691 IC50 = 8600 nM T21945 C7FBU8 44568693 IC50 = 7300 nM T21945 CD48SQ 44568694 IC50 = 1300 nM T21945 CSZ7V2 44568750 IC50 = 6000 nM T21945 CWG32I 44572166 Ki > 10000 nM T21945 C97VKX 44572751 Ki = 3404 nM T21945 CJ1VI8 44572802 Ki > 10000 nM T21945 CU25XD 44572810 Ki = 6780 nM T21945 CO1VA0 44574739 IC50 = 62 nM T21945 CIUN13 44574783 IC50 = 300 nM T21945 CO40XG 44574784 IC50 = 120 nM T21945 CX15IN 44574883 IC50 = 550 nM T21945 CX07AK 44574884 IC50 = 1100 nM T21945 C6S4IO 44576826 Ki = 3.4 nM T21945 C7WO9Z 44576828 Ki = 3.5 nM T21945 CE5JC1 44576830 Ki = 55 nM T21945 C4XBZ0 44576832 Ki = 49 nM T21945 COT0K9 44576862 Ki = 150 nM T21945 CYXV83 44576864 Ki = 75 nM T21945 CS4XT1 44576866 Ki = 31 nM T21945 CCB06N 44576868 Ki = 14 nM T21945 CV45DH 44576870 Ki = 230 nM T21945 C42FLK 44576888 Ki = 50 nM T21945 COP7S3 44576890 Ki = 430 nM T21945 C4ISW9 44576892 Ki = 2560 nM T21945 CC2GJ8 44578041 IC50 = 92 nM T21945 CS71BE 44578042 IC50 = 94 nM T21945 CHE5X2 44578075 IC50 > 322 nM T21945 C32VHN 44578076 IC50 = 300 nM T21945 CL2MG7 44578077 IC50 = 114 nM T21945 C4T5JW 44578112 IC50 > 400 nM T21945 CEO36B 44578113 IC50 > 400 nM T21945 CC0A8W 44578263 Ki = 70 nM T21945 CY40JQ 44578265 Ki = 27 nM T21945 CFJB16 44578266 Ki = 5 nM T21945 CE54ZK 44578267 Ki = 5 nM T21945 CSFE81 44578268 Ki = 7 nM T21945 CAQK40 44578269 Ki = 748 nM T21945 C5P0QK 44578270 Ki = 466 nM T21945 CQ30GC 44578271 Ki = 16 nM T21945 C8HB0Z 44578272 Ki = 29 nM T21945 CV63SW 44578313 Ki = 65 nM T21945 CH3U5D 44578314 Ki = 10 nM T21945 C8XAO4 44578315 Ki = 30 nM T21945 CS70JE 44578316 Ki = 86 nM T21945 CAP14F 44578317 Ki = 86 nM T21945 CUVQ89 44578318 Ki = 96 nM T21945 C17YVO 44578319 Ki = 8 nM T21945 CPQC54 44578368 Ki = 118 nM T21945 CA5I3W 44578369 Ki = 124 nM T21945 CTE6V8 44578370 Ki = 14 nM T21945 C4VO1L 44578371 Ki = 49 nM T21945 CXZ05B 44578372 Ki = 46 nM T21945 CVXD80 44578373 Ki = 89 nM T21945 C8AP4K 44578374 Ki = 23 nM T21945 CDMH40 44578375 Ki = 53 nM T21945 CUQV50 44579565 IC50 = 13 nM T21945 CS91HK 44579613 IC50 > 10 nM T21945 C0KBZ4 44580189 Ki > 2500 nM T21945 C2U7TG 44580702 Ki > 1000 nM T21945 C0S4IO 44580703 Ki > 1000 nM T21945 C3ONV6 44580704 Ki > 1900 nM T21945 C3L5ER 44583033 IC50 = 0.6 nM T21945 CBIO97 44585469 IC50 = 0.05 ug.mL-1 T21945 C4HJE6 44586246 Ki = 2880 nM T21945 CXKQ61 44587384 IC50 = 700 nM T21945 CZLV68 44587385 IC50 = 430 nM T21945 C8SFJ1 44587386 IC50 = 8000 nM T21945 CPBR52 44587387 IC50 = 140 nM T21945 C4D7GP 44587388 IC50 = 240 nM T21945 CRL0H9 44587389 IC50 = 45 nM T21945 C5PV7Q 44587390 IC50 = 14 nM T21945 C5IUL8 44587443 IC50 = 1300 nM T21945 C59KDV 44587445 IC50 = 3100 nM T21945 CLCE75 44587446 IC50 = 1000 nM T21945 CPF01B 44587447 IC50 = 420 nM T21945 CIL89C 44587448 IC50 = 370 nM T21945 CF0I6D 44587449 IC50 = 900 nM T21945 C0J4LS 44587450 IC50 = 27 nM T21945 CZVX16 44587463 IC50 = 5000 nM T21945 C6UI9D 44587464 IC50 = 4500 nM T21945 C6YQS2 44587465 IC50 = 30 nM T21945 CNV4I9 44587466 IC50 = 35 nM T21945 CL10BT 44587467 IC50 = 400 nM T21945 CX5KZ1 44587468 IC50 = 145 nM T21945 C0OYJ4 44587469 IC50 = 140 nM T21945 C2HUA1 44587470 IC50 = 180 nM T21945 CIW41M 44587471 IC50 = 75 nM T21945 CCKE83 44587472 IC50 = 15 nM T21945 C4SGR3 44587473 IC50 = 36 nM T21945 C47OBV 44587474 IC50 = 480 nM T21945 CQ79SU 44587475 IC50 = 9 nM T21945 CUE9C6 44587476 IC50 = 13 nM T21945 C37ZEB 44587477 IC50 = 11 nM T21945 CY0F1M 44587482 IC50 = 100 nM T21945 CL5M2J 44587483 IC50 = 370 nM T21945 CRN0Z1 44587484 IC50 = 1000 nM T21945 CTN0Q1 44587485 IC50 = 7 nM T21945 CAHW83 44587486 IC50 = 690 nM T21945 CJY60H 44587487 IC50 = 230 nM T21945 C3OL1M 44587488 IC50 = 39 nM T21945 C56QTZ 44587489 IC50 = 8 nM T21945 CD60KY 44587995 Ki = 1690 nM T21945 CZ98JO 44587997 Ki = 270 nM T21945 CAXU48 44587999 Ki = 160 nM T21945 C6FPZ9 44588001 Ki = 4100 nM T21945 C8F7IT 44588013 Ki = 180 nM T21945 C8LUE2 44588015 Ki > 5000 nM T21945 C7Y4QV 44588017 Ki = 2010 nM T21945 C5JQY4 44588019 Ki = 1230 nM T21945 C62JSH 44588021 Ki > 3000 nM T21945 C43ODT 44588187 Ki = 21.8 nM T21945 CKPE78 44588189 Ki = 1110 nM T21945 C57QYV 44588191 Ki = 330 nM T21945 CPR9K4 44588193 Ki = 2200 nM T21945 CLIV63 44588195 Ki = 1460 nM T21945 CN6RC7 44588197 Ki = 1850 nM T21945 CH18RV 44588223 Ki = 2710 nM T21945 CXA2D6 44588225 Ki = 2040 nM T21945 C4RZ1U 44588227 Ki = 2600 nM T21945 CQSC48 44588229 Ki > 3000 nM T21945 C4WB1N 44589201 Ki = 60 nM T21945 C69KAB 44590643 IC50 > 10000 nM T21945 CLQ2N4 44590644 IC50 > 10000 nM T21945 CJ2D4T 44590690 IC50 = 7983 nM T21945 C0RHT8 44590691 IC50 = 1774 nM T21945 CQCG57 44590692 IC50 = 628 nM T21945 CS7H9U 44590693 IC50 = 4746 nM T21945 C38PUH 44590694 IC50 = 481 nM T21945 CDB8Z5 44590725 IC50 = 3101 nM T21945 C0N5RO 44590726 IC50 = 2934 nM T21945 C4H6PT 44590727 IC50 = 2857 nM T21945 C3TUD7 44590728 Ki = 2222 nM T21945 CNL38Q 44590729 Ki = 4064 nM T21945 C7RBE8 44590819 Ki > 10000 nM T21945 CYBL93 44590820 Ki > 10000 nM T21945 CI6R1Z 44592120 IC50 = 6800 nM T21945 C1QO8J 44592121 IC50 = 10600 nM T21945 C7LKH8 44592122 IC50 > 10000 nM T21945 CVT6R5 44592123 IC50 = 40000 nM T21945 C04UVE 44592152 IC50 = 3000 nM T21945 C4KM6A 44592153 IC50 = 2600 nM T21945 CV8E7O 44592155 IC50 = 5600 nM T21945 CK47SV 44592156 IC50 = 3000 nM T21945 C4W1XJ 44592157 IC50 = 80 nM T21945 CMS5I2 44592158 IC50 = 5400 nM T21945 CSU06J 44592195 IC50 = 80 nM T21945 CZ6L3I 44592196 IC50 = 1500 nM T21945 CC52XI 44592242 IC50 = 827 nM T21945 CJO9K5 44592245 IC50 = 8400 nM T21945 CQ12YR 44593444 IC50 = 290 nM T21945 CPH6S0 44593451 IC50 = 7 nM T21945 C30HFZ 44593522 IC50 = 630 nM T21945 C1DI5Z 44593686 IC50 = 26 nM T21945 C7YLS4 44593687 IC50 = 26 nM T21945 C6KGF2 44593688 IC50 = 7 nM T21945 CU8F9L 44593689 IC50 = 200 nM T21945 CR18ZA 44593690 IC50 = 3 nM T21945 C20YZD 44593691 IC50 = 95 nM T21945 CN52LH 44593692 IC50 = 17 nM T21945 C7IU8S 44593694 IC50 = 5 nM T21945 C9SM4D 44593695 IC50 = 100 nM T21945 CSQ14O 44593696 IC50 = 7 nM T21945 CI10GR 44610722 IC50 = 735 nM T21945 CW84TH 44610723 IC50 = 2500 nM T21945 CPIB93 44610724 IC50 = 370 nM T21945 CVR29I 44625567 IC50 = 10 nM T21945 C24WVM 44625568 IC50 = 0.7943 nM T21945 COM81X 44625569 IC50 = 0.5012 nM T21945 CR8I3P 44625570 IC50 = 7.943 nM T21945 C2D0TJ 44625571 IC50 = 3.162 nM T21945 C6LD5P 44625653 IC50 = 1.995 nM T21945 C0A3WN 44626374 IC50 = 4 nM T21945 CR3PL6 44665680 Ki < 1000 nM T21945 CY47CM 45101948 IC50 = 800 nM T21945 CND19I 45102009 IC50 = 420 nM T21945 CW0RU3 45102635 EC50 = 28 nM T21945 CR83KY 45139778 IC50 = 9.7 nM T21945 CB16EP 45139780 IC50 = 4.6 nM T21945 C15AOE 45139782 IC50 = 72 nM T21945 CBDG89 45139784 IC50 = 14 nM T21945 C6ZL5S 45139960 IC50 = 23 nM T21945 CAKF28 45139962 IC50 = 2.3 nM T21945 C2RH4W 45139964 IC50 = 7.6 nM T21945 C10AOU 45139966 IC50 = 15 nM T21945 C1AWI8 45139968 IC50 = 170 nM T21945 CSC30M 45139970 IC50 = 2.6 nM T21945 CEB8M7 45139972 IC50 = 150 nM T21945 CHRV87 45140168 IC50 = 21 nM T21945 CO03PE 45140170 IC50 = 39 nM T21945 CO1KI6 45140172 IC50 = 5.7 nM T21945 C1S5GM 45140174 IC50 = 6.5 nM T21945 CXJ80R 45140176 IC50 = 19 nM T21945 CRW5G7 45140178 IC50 = 17 nM T21945 CXJ6A2 45140180 IC50 = 2.7 nM T21945 CT6XO9 45140370 IC50 = 1.4 nM T21945 CUOD26 45140371 IC50 = 3.7 nM T21945 C7MB5N 45141377 IC50 > 100 nM T21945 CMSH89 45141378 IC50 > 100 nM T21945 C05NYK 45141587 IC50 = 8.5 nM T21945 CTL0U6 45141609 IC50 > 100 nM T21945 CB9QZ6 45263405 IC50 = 19 nM T21945 CPGO97 45267145 IC50 = 4850 nM T21945 CTL3Z5 45267156 IC50 = 84 nM T21945 CT15YP 45267165 IC50 = 215 nM T21945 CZ3DW4 45267166 IC50 > 400 nM T21945 C5DGO1 45267167 IC50 = 35 nM T21945 CP7XE6 45267597 Ki = 60 nM T21945 CK58HY 45267611 Ki = 61 nM T21945 C3D9TN 45267621 Ki = 1258.93 nM T21945 CV1W8D 45267665 IC50 = 23 nM T21945 CEWR12 45268018 IC50 = 24 nM T21945 CD8G9N 45268026 IC50 > 400 nM T21945 CRP90V 45268466 Ki = 29 nM T21945 CSJ4L2 45268478 Ki = 28 nM T21945 CQJ9X1 45268495 Ki = 63.1 nM T21945 CO2X9T 45268882 IC50 = 45 nM T21945 C71XIB 45268898 IC50 = 42 nM T21945 CHP12M 45268914 IC50 = 3 nM T21945 CUQ23Z 45268922 IC50 = 43 nM T21945 C5OED7 45269318 Ki = 19 nM T21945 CF2P9H 45269325 Ki = 16 nM T21945 CQ03ZU 45269337 Ki = 30 nM T21945 CXE36D 45269351 Ki = 148 nM T21945 CVA9E0 45269726 IC50 = 13 nM T21945 CS0Z8C 45269735 IC50 = 23 nM T21945 CL6W3X 45269754 IC50 = 8 nM T21945 CX31KD 45270149 Ki = 294 nM T21945 C3GA6N 45270158 Ki = 10 nM T21945 C3KI7Q 45270163 Ki = 172 nM T21945 C0QR1E 45270171 Ki = 31 nM T21945 C6YI5N 45270172 Ki = 32 nM T21945 CZ9DA3 45270173 Ki = 18 nM T21945 C2M8FY 45270563 IC50 = 404 nM T21945 C13GPD 45270570 IC50 > 400 nM T21945 CM48NS 45270571 IC50 > 400 nM T21945 CH32XG 45270576 IC50 = 33 nM T21945 C0HV4C 45270577 IC50 = 23 nM T21945 COFD89 45270589 IC50 = 9 nM T21945 CEX26T 45270595 IC50 = 16 nM T21945 C13QSU 45270993 Ki = 22 nM T21945 CU9HV3 45271001 Ki = 18 nM T21945 C71AON 45271011 Ki = 43 nM T21945 CI01KJ 45271024 Ki = 794.33 nM T21945 C62UVG 45271383 IC50 = 91 nM T21945 C61TGI 45271390 IC50 = 23 nM T21945 C1S6TI 45271840 Ki = 72 nM T21945 C3QAP5 45271853 Ki = 37 nM T21945 CFG5Z3 45271864 Ki = 92 nM T21945 C3AJ7I 45271873 Ki = 199.53 nM T21945 CT04SP 45271883 Ki = 10 nM T21945 C1MKJ3 45272270 IC50 = 106 nM T21945 C1G9IK 45272302 IC50 = 9 nM T21945 CPM1U3 45272720 Ki = 19 nM T21945 C4VAE9 45272734 Ki = 38 nM T21945 C4P1FO 45273132 IC50 = 30 nM T21945 CUK91L 45273154 IC50 = 14 nM T21945 C5LB6F 45273161 IC50 = 48 nM T21945 C2DB0Y 45273169 IC50 > 400 nM T21945 CT3V0B 45273663 Ki = 24 nM T21945 CINR73 45273666 Ki = 572 nM T21945 C3Q0GZ 45273673 Ki = 825 nM T21945 CZU06K 45273676 Ki = 10 nM T21945 CQS5X0 45378248 Ki = 3.981 nM T21945 C7C9HW 45378386 Ki = 3.981 nM T21945 C51WBF 45378387 Ki = 3.981 nM T21945 CS04YD 45379827 Ki = 28.84 nM T21945 CMU6Z8 45379828 Ki = 1.738 nM T21945 C1SCJ9 45379829 Ki = 1288.25 nM T21945 CK6L2S 45379946 Ki = 1.95 nM T21945 CNQT48 45379947 Ki = 0.631 nM T21945 C5TQ8X 45379948 Ki = 125.89 nM T21945 CP82MH 45379949 Ki = 0.5012 nM T21945 CNSK69 45379950 Ki = 3.981 nM T21945 CM61UN 45380063 Ki = 158.49 nM T21945 C97ZQE 45380064 Ki = 12.59 nM T21945 CEFO86 45380065 Ki = 1.995 nM T21945 C53JYC 45380066 Ki = 39.81 nM T21945 C46FLB 45380180 Ki = 31.62 nM T21945 C89XTJ 45380181 Ki = 1.585 nM T21945 CYAE52 45380182 Ki = 316.23 nM T21945 C6BLR9 45380183 Ki = 1.995 nM T21945 CO8Z1P 45380184 Ki = 1 nM T21945 CE1M3S 45380185 Ki = 7.943 nM T21945 C1OK5Z 45481773 Ki = 515 nM T21945 CS0W9K 45481774 Ki > 10000 nM T21945 C5SN4D 45481775 Ki = 21 nM T21945 CZ02KA 45481776 Ki = 118 nM T21945 CCOL45 45481778 Ki = 960 nM T21945 CX68LG 45481779 Ki > 2000 nM T21945 C52FTP 45481780 Ki = 2000 nM T21945 C0NAE6 45481784 Ki > 2000 nM T21945 CG75XM 45481786 Ki = 1200 nM T21945 C5F8QK 45481787 Ki = 220 nM T21945 CQ89WZ 45481788 Ki > 2000 nM T21945 C7BQX4 45481789 Ki = 1170 nM T21945 C1O8ZD 45481790 Ki = 129 nM T21945 CO1Z4X 45481791 Ki = 1900 nM T21945 CF6R7M 45481792 Ki = 121 nM T21945 CWEK71 45481794 Ki = 690 nM T21945 C6SN1T 45483060 IC50 = 111 nM T21945 CJOP63 45483061 IC50 = 14 nM T21945 CMH54N 45483062 IC50 = 21 nM T21945 C6BP3U 45483063 IC50 = 15 nM T21945 COT26E 45483068 IC50 = 54 nM T21945 CDL5N0 45483069 IC50 = 21 nM T21945 C1OP5G 45483079 IC50 = 18 nM T21945 CQ4ZM0 45483080 IC50 = 16 nM T21945 C86FAI 45483083 IC50 = 304 nM T21945 C52YIE 45483084 IC50 = 22 nM T21945 CN50YU 45483087 IC50 = 527 nM T21945 CVL4X1 45483088 IC50 = 92 nM T21945 C5DZ3N 45483089 IC50 = 20 nM T21945 CY6Z9V 45483094 IC50 = 10 nM T21945 C8AY7V 45483095 IC50 = 11 nM T21945 CVY9K0 45483096 IC50 = 84 nM T21945 CZF8E4 45483097 IC50 = 232 nM T21945 CP7XI1 45483098 IC50 = 7 nM T21945 CQG68O 45483099 IC50 = 52 nM T21945 CS30CZ 45483103 IC50 = 64 nM T21945 C2S0EY 45483104 IC50 = 60 nM T21945 CCV7P6 45483105 IC50 = 124 nM T21945 CCF53Z 45483112 IC50 = 49 nM T21945 C4R6AY 45483113 IC50 = 21 nM T21945 CX3HT0 45483114 IC50 = 34 nM T21945 CYWX25 45483119 IC50 = 117 nM T21945 CCFO37 45483120 IC50 = 60 nM T21945 CRZ8V3 45483130 IC50 = 92 nM T21945 C97JBX 45483401 Ki = 1 nM T21945 C9K4XC 45483416 Ki = 2 nM T21945 CZQ6H8 45483429 Ki = 6 nM T21945 C3HAF8 45483430 Ki = 20 nM T21945 CG2SM9 45483458 Ki = 5 nM T21945 CFM9P8 45483465 Ki = 650 nM T21945 C5DS3M 45483506 Ki = 80 nM T21945 CHCA47 45483511 Ki = 192 nM T21945 C0HSJ7 45486515 IC50 = 415 nM T21945 C0IZ7C 45486517 IC50 = 79 nM T21945 C7E0XV 45486600 IC50 = 1200 nM T21945 C3HB5W 45486603 IC50 = 150 nM T21945 C0UV4I 45486616 IC50 = 1100 nM T21945 CR2J3T 45486621 IC50 = 42 nM T21945 CD8TC7 45486628 IC50 = 321 nM T21945 CMN6J2 45486630 IC50 = 118 nM T21945 COY84K 45486646 IC50 = 49 nM T21945 C8N6SO 45486651 IC50 = 230 nM T21945 CI89OX 45487689 IC50 = 1200 nM T21945 CC75GW 45487699 IC50 = 677 nM T21945 CNFI42 45487726 IC50 = 17400 nM T21945 CAO36Q 45487761 IC50 = 357 nM T21945 C80FMT 45487762 IC50 = 7000 nM T21945 CL9SM3 45487783 IC50 = 6000 nM T21945 CL1H2W 46200976 Ki = 632 nM T21945 C79ZBC 46200977 Ki = 406 nM T21945 CI39BE 46216792 IC50 > 10000 nM T21945 C34ZXM 46225029 Ki > 10000 nM T21945 CGY19F 46226540 Ki = 26 nM T21945 C79GDE 46226541 Ki = 4900 nM T21945 C0H7ID 46226542 Ki = 440 nM T21945 C5TSH8 46226543 Ki = 5400 nM T21945 CL07MO 46226544 Ki = 810 nM T21945 CMK1Z6 46226545 Ki = 180 nM T21945 C1KSD4 46226546 Ki = 100 nM T21945 CED57N 46226547 Ki = 2200 nM T21945 C27DWI 46226548 Ki = 1700 nM T21945 C3I4ZU 46226549 Ki = 1500 nM T21945 C6UDJ2 46226550 Ki = 5000 nM T21945 C8Q0JS 46226551 Ki = 1900 nM T21945 C6SGC5 46226552 Ki = 2700 nM T21945 C70RNJ 46226553 Ki = 3300 nM T21945 C72NRZ 46226554 Ki = 620 nM T21945 C8FM7G 46226555 Ki = 1300 nM T21945 CJS97C 46226556 Ki = 1200 nM T21945 CB8XA5 46226557 Ki = 120 nM T21945 COC3L5 46226572 Ki = 8.5 nM T21945 CJKZ16 46226573 Ki = 20 nM T21945 CF6I8D 46226574 Ki = 380 nM T21945 CE0W4J 46227268 IC50 = 2097 nM T21945 CY5FD9 46227269 IC50 = 2190 nM T21945 CJ9OF6 46228636 Ki = 0.5012 nM T21945 CSNI09 46228719 Ki = 19.95 nM T21945 CG68MR 46228720 Ki = 10 nM T21945 C5NB2Z 46228786 Ki = 7.943 nM T21945 C5JPE2 46229669 Ki = 1203 nM T21945 C4B0FX 46229670 Ki = 503 nM T21945 C39VDA 46229671 Ki = 8854 nM T21945 CS0EJ4 46229672 Ki = 667 nM T21945 C32VBR 46229686 Ki > 500 nM T21945 CN4HT2 46230756 Ki = 247 nM T21945 CI8O5W 46233622 IC50 = 6.2 nM T21945 C7OB2G 46235733 IC50 = 208.93 nM T21945 CJ2D3O 46701015 IC50 = 107.15 nM T21945 CM04ZI 46701016 IC50 = 95.5 nM T21945 C0JWP5 46701017 IC50 = 22.39 nM T21945 C5H0MJ 46701086 IC50 = 177.83 nM T21945 C9HWI7 46701087 IC50 = 204.17 nM T21945 CVE5O1 46701088 IC50 = 141.25 nM T21945 C1VPM0 46701089 IC50 = 56.23 nM T21945 CQ8B6R 46701090 IC50 = 38.02 nM T21945 C6C0FS 46701091 IC50 = 26.92 nM T21945 CC0M7T 46830494 IC50 = 2 nM T21945 C2ZGO0 46830791 IC50 = 4 nM T21945 CD0KX8 46831077 IC50 = 28 nM T21945 CYWA02 46831080 IC50 = 22 nM T21945 COF0Q6 46831083 IC50 = 25 nM T21945 CZF25N 46831086 IC50 = 51 nM T21945 CDF9H4 46831389 IC50 = 18 nM T21945 CL7XJ8 46831392 IC50 = 3 nM T21945 CEV89K 46831395 IC50 = 2 nM T21945 CC0OU8 46831694 IC50 = 36 nM T21945 CA2NE6 46832498 IC50 = 5 nM T21945 CCM24Q 46832501 IC50 = 602 nM T21945 C3J0YG 46832788 IC50 = 196 nM T21945 C02ASD 46832790 IC50 = 2255 nM T21945 CP4C2Q 46832792 IC50 = 9 nM T21945 C4K5MH 46832794 IC50 = 853 nM T21945 CJH2Y3 46832796 IC50 = 481 nM T21945 C8U6HQ 46833699 IC50 = 3 nM T21945 C95KSN 46833979 IC50 = 3 nM T21945 CV3CQ7 46833981 IC50 = 61 nM T21945 C18CYM 46833983 IC50 = 155 nM T21945 CUD7M8 46833985 IC50 = 143 nM T21945 CD0PH8 46833987 IC50 = 244 nM T21945 CHPS94 46833989 IC50 = 100 nM T21945 C80NHM 46834258 IC50 = 10 nM T21945 C1GPD3 46834260 IC50 = 6 nM T21945 C37MDG 46834262 IC50 = 277 nM T21945 CB75HC 46834537 IC50 = 2 nM T21945 CQ7S3X 46837648 IC50 = 32 nM T21945 CL7VN1 46837649 IC50 = 150 nM T21945 CU7OG4 46837651 IC50 = 3000 nM T21945 C5WNL1 46837652 IC50 = 1210 nM T21945 COX2H5 46837653 IC50 = 3800 nM T21945 CWZY17 46837780 IC50 = 830 nM T21945 CV2NT3 46837781 IC50 = 1680 nM T21945 CT83MU 46837782 IC50 > 100000 nM T21945 C5TY3Q 46837783 IC50 = 10300 nM T21945 CWJF83 46837784 IC50 = 740 nM T21945 C0ZSY5 46837785 IC50 = 151 nM T21945 CBQJ74 46837922 IC50 = 19 nM T21945 C8UWQ2 46837923 IC50 = 9 nM T21945 CCX8T0 46837924 IC50 = 170 nM T21945 CBH49N 46837925 IC50 = 527 nM T21945 CH76RQ 46855361 Ki = 63.1 nM T21945 CFJ3Q4 46855363 Ki = 1995.26 nM T21945 CEG23T 46855638 Ki = 19.95 nM T21945 CFW0B9 46855640 Ki = 7.943 nM T21945 CKS74N 46855641 Ki = 794.33 nM T21945 C7FPT6 46855642 Ki = 15.85 nM T21945 CZS2G8 46855643 Ki = 100 nM T21945 C9AG3X 46855785 Ki = 50.12 nM T21945 C2WKY8 46855786 Ki = 1258.93 nM T21945 CB51DQ 46855787 Ki = 1584.89 nM T21945 CHT1G5 46855789 Ki = 5011.87 nM T21945 CLX6M3 46855790 Ki = 63.1 nM T21945 C0CG4F 46866510 Ki = 3.981 nM T21945 C4X5GI 46879910 IC50 = 181.97 nM T21945 CK8A1O 46880462 Ki > 10000 nM T21945 C9KDP4 46880463 Ki > 10000 nM T21945 CODR73 46880498 Ki > 10000 nM T21945 CHJ5Y6 46880566 Ki > 10000 nM T21945 CE9PG2 46880567 Ki > 10000 nM T21945 C01PGO 46880568 Ki > 10000 nM T21945 CS7L4X 46880569 Ki > 10000 nM T21945 C0PXY7 46880628 Ki > 10000 nM T21945 CD37LU 46880629 Ki > 10000 nM T21945 CUY89F 46880630 Ki > 10000 nM T21945 C4P6XS 46880631 Ki > 10000 nM T21945 CJ53KF 46880672 Ki > 10000 nM T21945 CYJC08 46880673 Ki > 10000 nM T21945 C1RI9O 46880674 Ki > 10000 nM T21945 CU45MP 46881677 IC50 = 25 nM T21945 CMS27C 46882857 Ki = 10 nM T21945 CM45ZP 46882858 Ki = 11 nM T21945 C3IGF1 46882859 Ki = 198 nM T21945 CHLZ97 46882860 Ki = 43 nM T21945 C4B8EX 46882909 Ki = 103 nM T21945 CFY95C 46882910 Ki = 29 nM T21945 C6GJ1F 46882911 Ki = 67 nM T21945 C0SQX2 46882912 Ki = 139 nM T21945 CJ82WI 46882913 Ki = 26 nM T21945 CV94JW 46882937 Ki = 263 nM T21945 CM5Z4G 46882938 Ki = 65 nM T21945 CJV6R1 46882939 Ki = 169 nM T21945 C60YMF 46883462 Ki = 217 nM T21945 C7J6GU 46883497 Ki = 36 nM T21945 C3F5AS 46883498 Ki = 24 nM T21945 CRSE34 46883499 Ki = 13 nM T21945 C0CX3O 46883500 Ki = 37 nM T21945 C78FKZ 46888072 IC50 = 576 nM T21945 CH56AN 46890391 Ki = 22 nM T21945 CPDX34 46890392 Ki = 22 nM T21945 C0YGP2 46890393 Ki = 25 nM T21945 C61INJ 46890394 Ki = 340 nM T21945 CI14SE 46890441 Ki = 84 nM T21945 CP4GD3 46890442 Ki = 27 nM T21945 CQI2Y8 46890443 Ki = 58 nM T21945 CZ2MG7 46890444 Ki = 97 nM T21945 CP6A8K 46890445 Ki = 30 nM T21945 CD5J8B 46890446 Ki = 100 nM T21945 CYK9D2 46890489 Ki = 46 nM T21945 CCR04L 46890490 Ki = 26 nM T21945 CT4O9M 46890491 Ki = 40 nM T21945 CGPM19 46890493 Ki = 30 nM T21945 C68AJP 46933238 Ki = 1.259 nM T21945 CX7R3H 46933845 Ki > 10000 nM T21945 CAY75I 46934585 Ki = 3.162 nM T21945 C2LZJ0 49783209 Ki = 3226 nM T21945 C57SMG 49783415 Ki > 10000 nM T21945 C0TG6I 49783419 Ki > 10000 nM T21945 CO6W0D 49798171 Ki = 398.11 nM T21945 CHQ7I8 49798172 Ki = 501.19 nM T21945 CMBX16 49798173 Ki > 5011.87 nM T21945 CMO8V7 49798193 Ki = 50.12 nM T21945 C60YCR 49798194 Ki = 12.59 nM T21945 C85KNS 49798241 Ki = 1584.89 nM T21945 CQ4G1V 49798242 Ki = 316.23 nM T21945 C01JNE 49798243 Ki = 316.23 nM T21945 CC6MF8 49798244 Ki = 100 nM T21945 CYAS45 49798266 Ki = 316.23 nM T21945 C2UO0F 49799236 IC50 > 100000 nM T21945 C6FH8G 49799237 IC50 = 7950 nM T21945 CZ3US5 49799443 Ki = 501.19 nM T21945 CQH0U4 49799522 Ki = 63.1 nM T21945 CZ76MQ 49799633 IC50 = 114 nM T21945 CU28RO 49799634 IC50 = 2440 nM T21945 CN89XG 49799642 IC50 = 411 nM T21945 C85MBT 49799643 IC50 = 1570 nM T21945 CK6IA0 49799933 IC50 = 700 nM T21945 C58AWR 49818125 Ki = 0.07943 nM T21945 CDV79P 49818201 Ki = 1.413 nM T21945 CFX2Q0 49818202 Ki = 6.31 nM T21945 C23PXY 49818203 Ki = 3.162 nM T21945 CR40BA 49836386 IC50 = 0.22 nM T21945 C0M5XC 49836496 IC50 = 0.63 nM T21945 CZJV13 49852019 IC50 = 19 nM T21945 CSL8M9 49852020 IC50 = 0.9 nM T21945 CWCY74 49852021 IC50 = 6.3 nM T21945 CI08OL 49852022 IC50 = 14 nM T21945 C1BH4A 49852023 IC50 = 6.5 nM T21945 COR7M1 49863727 Ki = 2607 nM T21945 C7CJ5W 49863728 Ki = 142 nM T21945 C9YS5V 49863729 Ki = 87 nM T21945 CO3K6A 49863748 Ki = 145 nM T21945 CK92TE 49863749 Ki = 265 nM T21945 CFZ39O 49865822 Ki = 12.59 nM T21945 CT34HY 49865823 Ki = 158.49 nM T21945 CK7O1S 49865875 Ki = 7.943 nM T21945 CCH8T4 49865876 Ki = 2.512 nM T21945 C8V3NG 49865877 Ki = 2.512 nM T21945 CEK89Q 49865878 Ki = 12.59 nM T21945 CZA5X4 49865879 Ki = 7.943 nM T21945 CD4LO5 49865880 Ki = 7.943 nM T21945 CZ2W8K 49865881 Ki = 158.49 nM T21945 C0R8AN 49865934 Ki = 7.943 nM T21945 C9TN8D 49865935 Ki = 25.12 nM T21945 C3YJ4G 49865936 Ki = 3.162 nM T21945 CB5WR8 49865937 Ki = 1.995 nM T21945 C8LJ4H 49865983 Ki = 2.512 nM T21945 C1MPT6 49865984 Ki = 2.512 nM T21945 C62NWE 49865985 Ki = 3.162 nM T21945 C5H4AY 49865986 Ki = 0.631 nM T21945 C90XRC 49865987 Ki = 7.943 nM T21945 CKMX26 49866033 IC50 = 234 nM T21945 CEFJ14 49866038 Ki = 10 nM T21945 CZ9I3O 49866039 Ki = 5.012 nM T21945 C96XFK 49866040 Ki = 50.12 nM T21945 C26NLJ 49866041 Ki = 6.31 nM T21945 CQHM34 49866042 Ki = 0.5012 nM T21945 CK1Y3B 49866085 IC50 = 14.7 nM T21945 C8JY3K 49866095 Ki = 3.981 nM T21945 C9N5CZ 49866096 Ki = 10 nM T21945 CC1L4U 49866097 Ki = 2.512 nM T21945 CV49QI 49866161 Ki = 1.259 nM T21945 CF59UG 49866162 Ki = 19.95 nM T21945 C5N8KG 49866163 Ki = 1 nM T21945 C4F8UX 49866191 Ki = 7.943 nM T21945 C2RY0J 50878551 Ki < 10000 nM T21945 C2CYL1 50917604 Ki = 3855 nM T21945 C0C9HA 50917605 Ki = 29.1 nM T21945 C9U6BI 50917780 Ki = 16211 nM T21945 C6JNK5 50917781 Ki = 49.1 nM T21945 C1C9JT 50917784 Ki = 16877 nM T21945 C1BMO5 50917785 Ki = 66.2 nM T21945 C8J5MB 50941458 IC50 = 7141 nM T21945 CJP82R 50941459 IC50 = 926 nM T21945 CJ43IF 50941460 IC50 = 934 nM T21945 C2SHO8 50993865 IC50 = 73 nM T21945 CX48AD 51002362 Ki = 2129 nM T21945 C6LVM3 51003382 Ki = 116 nM T21945 CIW56N 51003383 EC50 = 97 nM T21945 CQ8KP7 51003749 IC50 = 15000 nM T21945 CE4KP1 51050257 Ki > 10000 nM T21945 CYR7P8 51346818 IC50 = 85 nM T21945 CD4B6S 51346820 IC50 = 295 nM T21945 CU2SX3 51355576 Ki = 250 nM T21945 CUQ53T 52918018 IC50 = 500 nM T21945 CTP6U5 52918019 IC50 = 16000 nM T21945 CL0BQ2 52945369 IC50 = 27 nM T21945 CJV4D0 52946564 IC50 = 26 nM T21945 C58FQG 52947784 IC50 = 3 nM T21945 CQCB97 52947785 IC50 = 11 nM T21945 C0K8CF 52947796 IC50 = 5 nM T21945 C8XB1M 52949040 IC50 = 12 nM T21945 C42NYA 53248999 Ki = 398.11 nM T21945 CGQJ07 53316788 Ki = 323 nM T21945 CR41UN 53316822 IC50 = 167 nM T21945 CL78NK 53316823 IC50 = 126 nM T21945 CB86XC 53316913 IC50 = 188 nM T21945 CE26AQ 53317143 IC50 = 9 nM T21945 C2V6WS 53317144 IC50 = 39 nM T21945 C9L6YK 53317145 IC50 = 63 nM T21945 CST69D 53317146 IC50 = 9990 nM T21945 CS9Z0R 53317167 IC50 = 269 nM T21945 CH76LD 53317168 IC50 = 10 nM T21945 C63XCS 53317410 IC50 = 60 nM T21945 C9RNL2 53317411 IC50 = 13 nM T21945 CZTW58 53317736 Ki = 528 nM T21945 CW70NZ 53318092 Ki = 489 nM T21945 C7PC1G 53318093 Ki = 1020 nM T21945 CQ37BK 53318094 Ki = 192 nM T21945 C8RLQ9 53318095 Ki = 1010 nM T21945 C85UKZ 53318218 IC50 = 54 nM T21945 CFHE24 53318434 IC50 = 6 nM T21945 CI49RQ 53318452 IC50 = 2188 nM T21945 CWHC74 53318453 IC50 = 28 nM T21945 CD0Y4B 53318705 IC50 = 891 nM T21945 CE1W5G 53318706 IC50 = 132 nM T21945 C8C7YZ 53318707 IC50 = 31 nM T21945 C8PAY5 53318980 IC50 = 3177 nM T21945 CZ0M8J 53319021 IC50 = 766 nM T21945 C8V1AW 53319232 IC50 = 1849 nM T21945 C5FRP2 53319428 Ki = 507 nM T21945 CY65NV 53319429 Ki = 164 nM T21945 C1MD0J 53319430 Ki = 374 nM T21945 C1E7BF 53319431 Ki = 1950 nM T21945 C2OJW5 53319432 Ki = 110 nM T21945 CT0W3X 53319433 Ki = 1140 nM T21945 C8EKT2 53319478 IC50 = 164 nM T21945 C79JCL 53319479 IC50 = 28 nM T21945 CK2G3D 53319480 IC50 = 210 nM T21945 CVXT03 53319481 IC50 = 372 nM T21945 C90TZS 53319482 IC50 = 1642 nM T21945 CJH1M0 53319767 IC50 = 232 nM T21945 CZ6L5C 53319784 IC50 = 232 nM T21945 CE6V4A 53319785 IC50 = 9217 nM T21945 C63JGV 53319832 IC50 = 23 nM T21945 CVF5U0 53319835 IC50 = 529 nM T21945 CXF1S4 53320328 IC50 = 72 nM T21945 CODA90 53320569 Ki = 5883 nM T21945 C19ZWJ 53320686 IC50 = 2597 nM T21945 CB84NG 53320778 IC50 = 117 nM T21945 C8JX4C 53320779 IC50 = 92 nM T21945 CP7RZ3 53320780 IC50 = 371 nM T21945 CL67KH 53320781 IC50 = 309 nM T21945 CK5C0S 53320864 IC50 = 19 nM T21945 CQ90IR 53321058 IC50 = 4 nM T21945 CZ7NM6 53321059 IC50 = 326 nM T21945 CXY92R 53321081 IC50 = 61 nM T21945 CS42VL 53321082 IC50 = 146 nM T21945 CO7L6Z 53321083 IC50 = 7 nM T21945 CSY1K4 53321125 IC50 = 960 nM T21945 CAJ4L7 53321331 IC50 = 90 nM T21945 CMZ7F8 53321332 IC50 = 5 nM T21945 C4X3IS 53321979 IC50 = 138 nM T21945 CLQ85U 53322027 Ki = 218 nM T21945 C53HJK 53322028 Ki = 328 nM T21945 CLD82J 53322084 IC50 = 27 nM T21945 C7QF2E 53322085 IC50 = 98 nM T21945 CY09UA 53322086 IC50 = 112 nM T21945 CBUT35 53322087 IC50 = 7262 nM T21945 CXL8W9 53322200 IC50 = 92 nM T21945 CE63PO 53322201 IC50 = 222 nM T21945 C3M9SC 53322397 IC50 = 19 nM T21945 CLT3Q2 53322398 IC50 = 36 nM T21945 CZLT60 53322409 IC50 = 26 nM T21945 CLZ41J 53322410 IC50 = 346 nM T21945 C3YWZ5 53322451 IC50 = 7 nM T21945 CZ92BF 53322452 IC50 > 10000 nM T21945 C5G8RQ 53322642 IC50 = 9 nM T21945 CRUF31 53322954 Ki = 1350 nM T21945 CND26W 53323338 IC50 = 1857 nM T21945 C6KAN9 53323339 IC50 = 3091 nM T21945 C2OB7G 53323389 Ki = 482 nM T21945 C4UBX5 53323390 Ki = 433 nM T21945 C1WU4E 53323391 Ki = 1000 nM T21945 CGN6Z3 53323531 IC50 = 26 nM T21945 CAQ07J 53323532 IC50 = 13 nM T21945 C1GZ3B 53323533 IC50 = 126 nM T21945 C4D1LX 53323761 IC50 = 114 nM T21945 CPKM07 53323762 IC50 = 790 nM T21945 CQW2S7 53323771 IC50 = 20 nM T21945 CO7TC1 53323812 IC50 = 5000 nM T21945 CDRV76 53323814 IC50 = 37 nM T21945 C32YWL 53324045 Ki = 518 nM T21945 C98OKX 53324333 IC50 = 206 nM T21945 C46XAC 53324366 IC50 = 1005 nM T21945 CR4W9L 53324553 Ki = 3623 nM T21945 CW58QL 53324656 IC50 = 1246 nM T21945 CFJ1B0 53324709 Ki = 73 nM T21945 C5I1FG 53324762 IC50 = 174 nM T21945 C94GOI 53324763 IC50 = 257 nM T21945 COP3J6 53324764 IC50 = 565 nM T21945 CE7DZ0 53324844 IC50 = 347 nM T21945 CB34ZM 53325028 IC50 = 22 nM T21945 CY9H2U 53325042 IC50 = 137 nM T21945 CRQF15 53325242 Ki = 77 nM T21945 C3QNR2 53325463 IC50 = 601 nM T21945 CZN8B4 53325581 IC50 = 45 nM T21945 COZ1W9 53325647 IC50 = 91 nM T21945 C1N7XO 53325966 IC50 = 1184 nM T21945 CZ69OW 53326010 Ki = 1640 nM T21945 CZ1U9T 53326011 Ki = 198 nM T21945 CM7YA0 53326118 IC50 = 12 nM T21945 CJ6G7X 53326119 IC50 = 67 nM T21945 CTH12B 53326554 IC50 = 85 nM T21945 C0M5WU 53391513 IC50 = 2454.71 nM T21945 C8DR9L 53391514 IC50 = 14125.38 nM T21945 C7GH1I 53391515 IC50 = 5888.44 nM T21945 C3BX4K 53391516 IC50 = 416.87 nM T21945 C5B1ST 53391517 IC50 = 537.03 nM T21945 CQYB97 53391614 IC50 = 6456.54 nM T21945 CK3D9F 53391615 IC50 > 10000 nM T21945 C3S5QX 53391616 IC50 > 10000 nM T21945 CI3T5Y 53391617 IC50 = 4265.8 nM T21945 CKOD62 53391618 IC50 = 208.93 nM T21945 CD24UN 53391714 IC50 = 190.55 nM T21945 CA0GN6 53391715 IC50 = 204.17 nM T21945 CQ4E2W 53391716 IC50 = 537.03 nM T21945 C64TJO 53391717 IC50 = 14.13 nM T21945 C3Q6IL 53391718 IC50 = 60.26 nM T21945 C7UBN1 53392848 IC50 = 2137.96 nM T21945 CB5JU8 53392849 IC50 = 4466.84 nM T21945 C0JI1M 53392850 IC50 = 3801.89 nM T21945 CPIT32 53392851 IC50 = 5370.32 nM T21945 C8K1TZ 53392852 IC50 = 2951.21 nM T21945 CS7TE6 53392939 IC50 = 912.01 nM T21945 CT7U5L 53392940 IC50 = 2344.23 nM T21945 CMOZ61 53475319 Ki = 436 nM T21945 CDV82B 53492877 IC50 = 5 nM T21945 CHE5Q4 54380151 Ki = 1400 nM T21945 CEY2B8 54583277 IC50 = 24 nM T21945 CF5Q0W 54583932 IC50 = 12000 nM T21945 C6ME0B 54584239 IC50 = 13 nM T21945 CY4F0W 54584873 IC50 = 28000 nM T21945 CL5I1R 54753271 Ki = 1350 nM T21945 CGO9V3 54756922 IC50 = 103 nM T21945 C4URA5 54756923 IC50 = 13 nM T21945 CYS19X 54756924 IC50 = 7 nM T21945 CLC71N 54756925 IC50 = 13 nM T21945 CF82MX 54756926 IC50 = 207 nM T21945 CY7IR2 54757020 IC50 = 199 nM T21945 CT5F4Z 54757021 IC50 = 5 nM T21945 CPW0G4 54757022 IC50 = 8 nM T21945 CYX2L8 54757023 IC50 = 120 nM T21945 CCZ97U 54757024 IC50 = 7 nM T21945 COJ0T5 54757025 IC50 = 5 nM T21945 C13SMB 54757119 IC50 = 99 nM T21945 CGT6F0 54757120 IC50 = 611 nM T21945 C4S6UM 54757121 IC50 = 199 nM T21945 CP5S0U 54757122 IC50 = 80 nM T21945 CYB78R 54757668 Ki = 2900 nM T21945 CL75BS 54765676 IC50 = 327.9 nM T21945 CB87MF 54766009 IC50 = 205.7 nM T21945 C93WMS 54767239 IC50 = 427.6 nM T21945 CLV3N6 54767240 IC50 = 477.5 nM T21945 CZ47UJ 54767241 IC50 = 68.9 nM T21945 C5RX1P 54767242 IC50 = 633.5 nM T21945 C32NWX 54767413 IC50 = 249.9 nM T21945 C6ASW2 54767576 IC50 = 495 nM T21945 C45SEW 54767744 IC50 = 1456.3 nM T21945 C3KV8R 54767747 IC50 = 2541.5 nM T21945 CO6CJ2 54767906 IC50 = 373.5 nM T21945 CMJ32F 56659126 Ki = 39.81 nM T21945 CQ6XM7 56659146 Ki = 39.81 nM T21945 CFT9V8 56659147 Ki = 25.12 nM T21945 CO0GR7 56659199 Ki = 0.3981 nM T21945 CC26HR 56659200 Ki = 31.62 nM T21945 CGID30 56659201 Ki = 1.585 nM T21945 CG0M7T 56662629 Ki = 50.12 nM T21945 CP2ZS4 56662647 Ki = 63.1 nM T21945 C8NIZ3 56662648 Ki = 50.12 nM T21945 CN7WB5 56662696 Ki = 50.12 nM T21945 CD9F3J 56662697 Ki = 25.12 nM T21945 C5HF9D 56666091 Ki = 19.95 nM T21945 C9RE3V 56669493 Ki = 10 nM T21945 CK3R7P 56669494 Ki = 100 nM T21945 CVRH79 56669561 Ki = 0.631 nM T21945 CC9XR7 56669562 Ki = 3.162 nM T21945 CXE9A8 56669563 Ki = 1 nM T21945 CU0NE5 56672197 Ki > 10000 nM T21945 CNK39V 56673078 Ki = 6.31 nM T21945 C93KBW 56679646 Ki = 10 nM T21945 CAR8M5 56679647 Ki = 39.81 nM T21945 CN1C3K 56679724 Ki = 31.62 nM T21945 CP3L7E 56682094 Ki > 10000 nM T21945 CET3N2 56682964 Ki = 19.95 nM T21945 CK73UC 56683046 Ki = 0.3981 nM T21945 CZR91E 56683047 Ki = 39.81 nM T21945 C60IBF 56683048 Ki = 10 nM T21945 CJKO58 56852956 Ki = 2754.23 nM T21945 C73MZW 56924689 IC50 = 4400 nM T21945 C90DOS 56942993 IC50 = 93 nM T21945 CHN2F6 56949640 Ki = 191 nM T21945 CZI53T 56961001 IC50 = 5.6 nM T21945 C1TC7Q 56963799 Ki > 10000 nM T21945 CBO89M 57384807 IC50 = 960 nM T21945 C2BAZ9 57385041 IC50 = 1300 nM T21945 C2TAS4 57385549 IC50 = 880 nM T21945 CX2TG9 57385550 IC50 = 2400 nM T21945 CVM67R 57385790 IC50 = 760 nM T21945 CCJ93V 57391031 Ki = 12090 nM T21945 C9LX1S 57391709 Ki = 188 nM T21945 C6SZ4E 57396296 Ki = 27.7 nM T21945 C6HBG0 57396813 IC50 = 4400 nM T21945 CX0B5M 57403525 Ki = 1225 nM T21945 C4N3VY 57403918 Ki = 426 nM T21945 CHU5T7 57523687 EC50 = 1760 nM T21945 C0WJ4E 58954830 IC50 = 17 nM T21945 CSF52J 58954867 IC50 = 3 nM T21945 C9ZP3D 58954900 IC50 = 23 nM T21945 CHQE32 58954945 IC50 = 943 nM T21945 CK6W7I 59536635 IC50 = 6.9 nM T21945 CI5PM3 60165413 Ki = 49 nM T21945 C3K5JN 60165681 Ki > 10000 nM T21945 CGF3J5 66572162 IC50 = 327 nM T21945 CZL90M 66572393 IC50 = 385 nM T21945 C2UZ3A 66572397 IC50 = 265 nM T21945 CCR2I5 66572399 IC50 = 178 nM T21945 C35VKU 66572510 IC50 = 531 nM T21945 CL8R5V 66975152 IC50 = 0.21 nM T21945 C0OC8T 66975291 IC50 = 2.3 nM T21945 CCN1W5 66975591 IC50 = 0.079 nM T21945 C23DPF 66975638 IC50 = 0.77 nM T21945 C3W0XI 66975648 IC50 = 52 nM T21945 C51JHP 66975671 IC50 = 5.8 nM T21945 CV19LA 66975764 IC50 = 0.1 nM T21945 C50HKX 66975948 IC50 = 5.8 nM T21945 C0L2QJ 66976018 IC50 = 700 nM T21945 CE9A4J 66976134 IC50 = 1.1 nM T21945 CZE5S6 66976296 IC50 = 0.13 nM T21945 C78MWK 66976356 IC50 = 0.64 nM T21945 C5EM9P 66976389 IC50 = 12 nM T21945 CP3M9I 66976532 IC50 = 0.33 nM T21945 CAL40U 66976565 IC50 = 0.065 nM T21945 CI29HX 66976607 IC50 = 0.08 nM T21945 C6I7SV 66976613 IC50 = 2 nM T21945 C8LD7M 66976718 IC50 = 17 nM T21945 C6ON5Y 66976777 IC50 = 13 nM T21945 CB05ID 67972431 EC50 = 339 nM T21945 C0MYB6 68653619 Ki = 250 nM T21945 CNY0W5 68673707 IC50 = 55 nM T21945 C76ROM 68673872 IC50 = 33 nM T21945 CSF80C 68993720 IC50 = 69 nM T21945 CVZ51D 68993987 IC50 < 1 nM T21945 CN0MY2 68994312 IC50 = 5 nM T21945 CKTA56 68994365 IC50 = 5.2 nM T21945 CE1WF3 68994389 IC50 = 2.9 nM T21945 CN08VY 68994725 IC50 = 16 nM T21945 C0ZY9I 68994988 IC50 = 23 nM T21945 CR3H9X 68995479 IC50 = 11 nM T21945 C1LWS9 68995587 IC50 = 180 nM T21945 CDLR80 68995667 IC50 = 6 nM T21945 CCIV97 68995742 IC50 = 1.3 nM T21945 C2MK1S 68995928 IC50 = 15 nM T21945 C56VJS 68996260 IC50 = 2.6 nM T21945 CQ4Y2V 68996331 IC50 = 22 nM T21945 CHI19N 68996402 IC50 = 8.8 nM T21945 C17BRZ 68997664 IC50 = 5.5 nM T21945 CDT9Z5 68998740 IC50 = 1000 nM T21945 CP0AR5 68999429 IC50 = 41 nM T21945 CN14QD 69000395 IC50 < 3 nM T21945 CNM1U4 69397184 Ki = 35 nM T21945 CYM94S 70676472 IC50 = 10 nM T21945 C7J0FD 70676474 IC50 = 12 nM T21945 CLTA38 70676476 IC50 = 3.1 nM T21945 CMN57J 70676478 IC50 = 16 nM T21945 C9QZ7C 70676480 IC50 = 21 nM T21945 C7W3JA 70681326 Ki = 12.59 nM T21945 C67CHV 70681491 Ki > 10000000 nM T21945 C39QGY 70683608 Ki > 10000000 nM T21945 C60SBP 70685515 Ki = 199.53 nM T21945 CCOR65 70685727 Ki = 5454000 nM T21945 C3UO2F 70686000 IC50 = 1000 nM T21945 C1CH5A 70687667 Ki = 1000 nM T21945 CWO02R 70688127 IC50 = 1700 nM T21945 CTVW13 70689263 Ki = 4340 nM T21945 C7RA0K 70689264 Ki = 1120 nM T21945 CKMJ68 70689265 Ki = 2800 nM T21945 C59NVG 70691872 IC50 = 0.3981 nM T21945 CB3NW6 70693452 Ki = 2920 nM T21945 CP38FE 70693453 Ki = 390 nM T21945 C8IQC6 70695563 Ki = 222 nM T21945 C5DP3J 70695564 Ki = 136 nM T21945 C37USC 70697274 Ki = 503 nM T21945 CKD60A 70789640 Ki = 1289 nM T21945 CI93FE 70963695 IC50 = 3200 nM T21945 C2FN8M 71134973 IC50 = 2.1 nM T21945 C5BER9 71332336 IC50 = 5328 nM T21945 C9VZ8J 71450550 Ki = 9905 nM T21945 C5X3LM 71450608 Ki = 806 nM T21945 C87FQH 71450609 Ki = 29 nM T21945 C4TWS5 71452172 Ki = 203 nM T21945 C4NDR3 71452382 Ki > 10000 nM T21945 C6G2HC 71455894 Ki > 10000 nM T21945 C7MNB5 71457264 Ki = 2006 nM T21945 C6X1GN 71457767 Ki = 7.1 nM T21945 C87FDI 71458022 IC50 > 10 nM T21945 CK5T4P 71459604 Ki = 3638 nM T21945 CD3L7R 71463125 Ki = 115 nM T21945 C4RAQ6 71518063 Ki = 11800 nM T21945 CO26TC 71541094 Ki = 74 nM T21945 CE8YO0 71541095 Ki = 130 nM T21945 CN79ZY 71541096 Ki = 12 nM T21945 CNCR14 71541097 Ki = 15 nM T21945 CW34SU 71541098 Ki = 57 nM T21945 CKW24J 71541099 Ki = 12 nM T21945 C0ZL6O 71541186 Ki = 54 nM T21945 C92PZK 71541187 Ki = 130 nM T21945 C0T4RD 71541188 Ki = 120 nM T21945 CB91FO 71541189 Ki = 66 nM T21945 CY5E0J 71541190 Ki = 17 nM T21945 C4XK1S 71541191 Ki = 24 nM T21945 C32HNI 71541192 Ki = 25 nM T21945 C9C0JU 71541193 Ki = 83 nM T21945 CFO05K 71541194 Ki = 170 nM T21945 CD1T5J 71541195 Ki = 130 nM T21945 CBWZ86 71541287 Ki = 250 nM T21945 CK82YE 71541288 Ki = 430 nM T21945 CQ81HF 71541289 Ki = 46 nM T21945 CU53JE 71541292 Ki = 4 nM T21945 C57KER 71541293 Ki = 430 nM T21945 C6B3CF 71562265 IC50 = 0.3981 nM T21945 C9V0FZ 71562266 IC50 = 5.012 nM T21945 C49VSK 71562370 IC50 = 3.162 nM T21945 COFY97 71562371 IC50 = 7.943 nM T21945 C1JCZ5 71562372 IC50 = 0.7943 nM T21945 CXR0E7 71562373 IC50 = 3.981 nM T21945 C4PDM8 71562374 IC50 = 10 nM T21945 C3L9HK 71562375 IC50 = 1.995 nM T21945 CX7VK3 71562376 IC50 = 0.5012 nM T21945 CHW7K1 71562377 IC50 = 31.62 nM T21945 CK95GV 71562472 IC50 = 5.012 nM T21945 C4NS5W 71562473 IC50 = 3.981 nM T21945 C6X9SM 71562474 IC50 = 50.12 nM T21945 C1H4KQ 71562475 IC50 = 10 nM T21945 C6X3BP 71562476 IC50 = 0.5012 nM T21945 CH49FE 71562477 IC50 = 1.585 nM T21945 CU1CZ6 71562478 IC50 = 0.7943 nM T21945 CPAY18 71562479 IC50 = 1.995 nM T21945 CY39RM 71562586 IC50 = 0.3981 nM T21945 C4F2UW 71562587 IC50 = 1.995 nM T21945 CI3KA2 71562588 IC50 = 5.012 nM T21945 C13NIO 71562589 IC50 = 0.7943 nM T21945 CKPH80 71562590 IC50 = 3.981 nM T21945 C0NIA6 71562591 IC50 = 1.995 nM T21945 CRCT65 71562592 IC50 = 0.5012 nM T21945 C1XQ5M 71562593 IC50 = 31.62 nM T21945 CFQP86 71562712 IC50 = 5.012 nM T21945 CPDV40 71562713 IC50 = 3.981 nM T21945 CP2N3Y 71562714 IC50 = 50.12 nM T21945 CS59VG 71562715 IC50 = 10 nM T21945 CE7X9R 71562716 IC50 = 0.5012 nM T21945 CP20LV 71562717 IC50 = 1.259 nM T21945 CQU78X 71562718 IC50 = 0.631 nM T21945 CCO48Y 71562719 IC50 = 1 nM T21945 CSYR25 71562833 IC50 = 0.3162 nM T21945 CF0R4S 71562834 IC50 = 3.981 nM T21945 C5NO2C 71562835 IC50 = 3.981 nM T21945 C2UQD4 71562836 IC50 = 0.7943 nM T21945 C1Q4JZ 71562837 IC50 = 1.585 nM T21945 CZWN24 71716486 IC50 = 2.512 nM T21945 CH8O3Z 71717705 IC50 = 5.012 nM T21945 C0O4ID 71718185 Ki = 5.1 nM T21945 C7TCH6 71718282 Ki = 194 nM T21945 CM7T0H 71719533 IC50 = 1 nM T21945 C2EWG5 71719830 Ki = 49 nM T21945 CY6DR8 71727648 IC50 = 25 nM T21945 CA3H0X 71727754 IC50 = 110 nM T21945 C2WD4V 71727756 IC50 = 28 nM T21945 CDT2P5 71727758 IC50 = 9.3 nM T21945 C39EUA 71727760 IC50 = 8.7 nM T21945 C8BLG9 71727762 IC50 = 200 nM T21945 C1XB7U 71727764 IC50 = 18 nM T21945 CS83FB 71727766 IC50 = 12 nM T21945 CX7O8K 71727768 IC50 = 14 nM T21945 CEM15Z 71727886 IC50 = 44 nM T21945 C5BL4F 71727888 IC50 = 28 nM T21945 CX21QS 71727890 IC50 = 22 nM T21945 COUT12 71812204 IC50 = 15 nM T21945 CT03WY 72202713 IC50 = 865.7 nM T21945 CKS1Z3 72202714 IC50 = 509.5 nM T21945 CIR13D 72202716 IC50 = 3825 nM T21945 CR5Q0P 72202718 IC50 = 7619 nM T21945 CTL7Z6 72202847 IC50 = 2521 nM T21945 C1UO9J 72202848 IC50 = 1662 nM T21945 CJ7VK8 72202849 IC50 = 2745 nM T21945 C4V2NE 72202850 IC50 = 1900 nM T21945 CDG0A8 72202852 IC50 = 1187 nM T21945 CV5TJ6 72202983 IC50 = 482.9 nM T21945 C3ZHJ1 72202984 IC50 = 990.3 nM T21945 CS3B7C 72202985 IC50 = 1376 nM T21945 CWH6T3 72548703 IC50 = 3.4 nM T21945 C48RGH 72737188 Ki = 785 nM T21945 CAEQ04 72737189 Ki = 153 nM T21945 CC65OA 73213195 Ki = 1348.96 nM T21945 CW83DK 73213196 Ki = 1949.84 nM T21945 C6J0TM 73346336 Ki = 8533 nM T21945 CK48PN 73347369 Ki = 177 nM T21945 C4YV6S 73347524 IC50 = 120 nM T21945 CEQS50 73347526 IC50 = 130 nM T21945 CI0JV6 73347528 IC50 = 70 nM T21945 C85LKM 73348886 Ki = 1.2 nM T21945 C9Y6OD 73348887 Ki = 438 nM T21945 CM50LN 73349057 IC50 = 36 nM T21945 C7XOF4 73349320 IC50 = 2033 nM T21945 CT69RQ 73349828 Ki = 56 nM T21945 C5RSW2 73349830 Ki = 3.2 nM T21945 C75HSZ 73350217 EC50 = 1380.38 nM T21945 CHNT68 73350623 IC50 = 21 nM T21945 CRL1C0 73351722 EC50 = 1819.7 nM T21945 C68XHC 73353199 IC50 = 25000 nM T21945 CCD70L 73353582 IC50 = 98 nM T21945 C7BMX2 73353673 Ki = 867 nM T21945 C1NJ0R 73353884 Ki = 7352 nM T21945 CYPL06 73355375 IC50 = 384.2 nM T21945 CWK70C 73356510 Ki = 30 nM T21945 C50CMV 76309752 Ki = 1810 nM T21945 C1Y9WZ 76316965 Ki = 8250 nM T21945 CJX71S 76320688 Ki = 259 nM T21945 C8YW4N 76324331 Ki = 7580 nM T21945 CP1U7E 76327897 Ki = 5580 nM T21945 C8S1PB 76327898 Ki = 2920 nM T21945 C1WZ5N 76331540 Ki = 3170 nM T21945 C47EDP 76331541 Ki = 997 nM T21945 C5N6LG 76331542 Ki = 8410 nM T21945 C2QWJ5 76335158 Ki = 577 nM T21945 C4G6RW 76335160 Ki = 3550 nM T21945 CM54ZS 76335161 Ki = 1630 nM T21945 C2LQ5Z 89437491 IC50 = 136.4 nM T21945 CP29UR 89838714 IC50 = 6 nM T21945 CF6P3I 89843681 IC50 = 8.5 nM T21945 CBH87U 91667621 IC50 = 6 nM T21945 C0RV4M 91799659 IC50 = 3.8 nM T21945 CCY0O2 100951644 IC50 = 5300 nM T21945 C10DAF 112777136 IC50 = 129800 nM T21945 C7AYV5 118540795 Ki = 3160 nM T21945 CA79GZ 118706038 IC50 = 33.5 nM T21945 CGBC58 118706039 IC50 = 37.2 nM T21945 C5LCJ1 118706532 IC50 = 33.7 nM T21945 CI2FN5 118706536 IC50 = 10.6 nM T21945 C2BG1F 118706537 IC50 = 30 nM T21945 C2WP6X 118706538 IC50 = 15.9 nM T21945 CZE4U0 118706539 IC50 = 14.6 nM T21945 CX8I0G 118706540 IC50 = 32.5 nM T21945 C4S9VT 118706541 IC50 = 30.8 nM T21945 CKD94F 118706542 IC50 = 68.6 nM T21945 C0KQO9 118706543 IC50 = 14.7 nM T21945 C5HJY0 118706544 IC50 = 33.1 nM T21945 CJ15AS 118708361 IC50 = 13 nM T21945 C7XEC0 118708362 IC50 = 260 nM T21945 CK30WF 118708364 IC50 = 2000 nM T21945 CG7W4D 118708365 IC50 = 660 nM T21945 C6UJC5 118708366 IC50 = 1700 nM T21945 CLQ52I 118708373 IC50 = 570 nM T21945 CSB25E 118709750 Ki = 510 nM T21945 CD4S9R 118709751 Ki = 462 nM T21945 CD34IY 118710582 IC50 = 8.3 nM T21945 CD1O7G 118710583 IC50 = 9100 nM T21945 C05FSJ 118714012 IC50 = 157.3 nM T21945 CY6AF2 118714015 IC50 = 635.4 nM T21945 C15FVH 118714017 IC50 = 425.7 nM T21945 CGC5J6 118719847 IC50 = 82 nM T21945 C6HV3B 118730351 EC50 = 1180 nM T21945 C3LZM9 118730352 EC50 = 670 nM T21945 CS7HB2 118871454 IC50 = 420100 nM T21945 CDU18K 118871456 IC50 = 687200 nM T21945 C1Z4TP 118871458 IC50 = 108200 nM T21945 CQ8H1J 118871471 IC50 = 174000 nM T21945 CSC5J4 121488665 Ki = 227 nM T21945 CUK9E2 122181877 IC50 = 3.3 nM T21945 CHKY46 122181879 IC50 = 3.4 nM T21945 CR5ES2 122188495 IC50 = 267 nM T21945 C5Y2LX 122188496 IC50 = 268 nM T21945 CG6UW3 122188497 IC50 = 621 nM T21945 C12TIS 122188498 IC50 = 4750 nM T21945 CL7PH5 122188499 IC50 = 153 nM T21945 C9TDA7 122188500 IC50 = 2020 nM T21945 CARF60 122188503 IC50 = 340 nM T21945 CC87DN 122188504 IC50 = 885 nM T21945 CQZ0A3 122188505 IC50 = 238 nM T21945 C1CJQ0 122188571 EC50 = 900 nM T21945 C8L1FV 122188773 IC50 = 472 nM T21945 CJ6G5D 122188774 IC50 = 1680 nM T21945 CNT50I 122188775 IC50 = 8030 nM T21945 CA8QW0 122188776 IC50 = 275 nM T21945 C8K9XA 122196341 IC50 > 1200 nM T21945 CM57GR 126720252 Ki = 1870 nM T21945 CTBN56 127026052 Ki = 1995.26 nM T21945 CEJ3R5 127029340 IC50 = 33 nM T21945 C6H5KN 127030249 IC50 = 2500 nM T21945 CCD8P5 127032017 IC50 = 2100 nM T21945 CQS75W 127032626 IC50 = 1070 nM T21945 CX6J8Y 127033284 IC50 = 530 nM T21945 CY82JA 127033285 IC50 = 610 nM T21945 CU8K1Q 127033286 IC50 = 760 nM T21945 C1ZMH0 127033287 IC50 = 1170 nM T21945 C0YF3E 127033288 IC50 = 560 nM T21945 C3IPX2 127033888 IC50 = 600 nM T21945 CF3XL5 127033889 IC50 = 890 nM T21945 C5QGV3 127033890 IC50 = 380 nM T21945 CQ0ZT9 127035062 Ki = 11 nM T21945 CU49VE 127036186 Ki < 10000 nM T21945 CG06BD 127036932 Ki = 630.96 nM T21945 CVW71O 127036953 Ki = 1000 nM T21945 CWJ59Z 127051882 IC50 = 1.4 nM T21945 C1RI8Q 132060720 Ki = 100 nM T21945 C4OC0I 132060752 Ki = 1312 nM T21945 CGHO19 132060770 Ki = 1059 nM T21945 CXV95T 132578504 IC50 = 500 nM T21945 C8NUR9 132578505 IC50 = 460 nM T21945 CGW0I7 132578506 IC50 = 800 nM T21945 CI4OC9 132578507 IC50 = 670 nM T21945 C5GEB2 132578508 IC50 = 510 nM T21945 C3ONX2 132578509 IC50 = 1620 nM T21945 CAVB41 132584404 Ki > 10000 nM T21945 CBU81N 134149168 Ki > 10000 nM T21945 C1GY2T 135156251 EC50 > 10000 nM T21945 C3QOP1 136340699 IC50 = 1 nM T21945 C4UON5 136389176 IC50 = 1.9 nM T21945 CG05IL 136389183 IC50 = 100 nM T21945 CP0E8J 136389204 IC50 = 25 nM T21945 C2QCA5 137631487 EC50 = 1520 nM T21945 CF3ZY7 137631557 IC50 = 85700 nM T21945 C5XL1N 137631893 Ki = 70 nM T21945 C14RKA 137632704 IC50 = 112600 nM T21945 C0C6ZL 137632750 IC50 = 1350 nM T21945 CCP46O 137633241 IC50 = 57600 nM T21945 C5G0XW 137633601 EC50 = 310 nM T21945 C8HPN4 137634334 EC50 = 65 nM T21945 C2LJW0 137634948 IC50 = 3450 nM T21945 CR74SC 137635327 IC50 = 568.9 nM T21945 CW9X5R 137635426 IC50 = 1327 nM T21945 CX17BR 137635648 IC50 = 3030 nM T21945 C42HCS 137636472 IC50 = 3000 nM T21945 CKQ92P 137636703 IC50 = 2280 nM T21945 COH18X 137637663 IC50 = 152500 nM T21945 CL56ZQ 137637671 IC50 = 1260 nM T21945 CD31YG 137638231 IC50 = 2510 nM T21945 C1EU5S 137638283 IC50 = 5020 nM T21945 CJI0K6 137638828 EC50 = 740 nM T21945 CBK0I8 137639266 EC50 = 400 nM T21945 C4BXH9 137640164 IC50 = 227500 nM T21945 CV20BW 137640543 IC50 = 5860 nM T21945 CVC6R8 137640624 IC50 = 519 nM T21945 C1X0QZ 137640906 IC50 = 2580 nM T21945 C06KGS 137641034 IC50 = 3080 nM T21945 CE8N4S 137641762 Ki = 3100 nM T21945 C70XZQ 137643636 EC50 = 26 nM T21945 C9VR5M 137643839 IC50 = 1313 nM T21945 CASM14 137643954 IC50 = 144200 nM T21945 C3ZRY2 137645338 IC50 = 5100 nM T21945 CPCY48 137645406 Ki = 931 nM T21945 C85OYG 137645602 IC50 = 99 nM T21945 C1KT5F 137645761 IC50 = 4340 nM T21945 CPZ3E1 137646230 IC50 = 329 nM T21945 CE6NB3 137646374 IC50 = 145800 nM T21945 CT7UG4 137646579 IC50 = 30000 nM T21945 CE9M3Z 137648195 IC50 = 3750 nM T21945 CIH3O8 137648265 IC50 = 2830 nM T21945 CL06NY 137648464 EC50 = 627 nM T21945 C0EVB7 137648614 IC50 = 318 nM T21945 CG1ME5 137648669 IC50 = 3960 nM T21945 CUFO39 137649223 EC50 = 251 nM T21945 CO4VY9 137649584 IC50 = 188100 nM T21945 C6YE5R 137649990 IC50 = 67200 nM T21945 C6GL0F 137652257 IC50 = 521 nM T21945 C65XKJ 137653127 EC50 = 254 nM T21945 CR9F3Q 137653203 EC50 = 1520 nM T21945 C02HUF 137653618 IC50 > 10000 nM T21945 CR25WM 137653998 EC50 = 490 nM T21945 C1JGO6 137654323 IC50 = 4218 nM T21945 CT35OC 137654501 IC50 = 3460 nM T21945 C96BJN 137654642 IC50 = 1590 nM T21945 C46UFA 137654647 IC50 = 5520 nM T21945 CF7M8V 137655321 IC50 = 1467 nM T21945 C3LG7W 137655838 EC50 = 1390 nM T21945 CU3DK5 137655842 IC50 = 1710 nM T21945 CZ84KG 137656433 IC50 = 323 nM T21945 CN2UE9 137656598 EC50 = 827 nM T21945 CQ1SI8 137656684 IC50 = 1621 nM T21945 CZ1XS0 137656786 IC50 = 68400 nM T21945 C56MCJ 137656979 EC50 = 980 nM T21945 C3GX2Z 137657462 IC50 = 71000 nM T21945 CSA8G2 137658186 IC50 = 767500 nM T21945 CG92PT 137660066 IC50 = 1530 nM T21945 CWX6N4 137660247 IC50 = 3000 nM T21945 CEV40N 137661034 IC50 = 1760 nM T21945 CLF7V1 137661266 IC50 = 1323 nM T21945 CCSU34 137661732 IC50 = 3590 nM T21945 CS47KN 137662116 IC50 = 399.5 nM T21945 C4E5ZX 141363479 IC50 > 10000 nM T21945 COT18S 145011254 Ki > 10000 nM T21945 C9A1VD 145967813 IC50 = 3.2 nM T21945 CM8TF3 145968603 Ki = 50.12 nM T21945 C4BS6T 145969809 IC50 = 10 nM T21945 CUQ7E0 145970103 Ki = 3.981 nM T21945 CBT6L8 145970391 IC50 = 2 nM T21945 CF67IA 145970695 Ki = 79.43 nM T21945 CB7O9W 145971077 Ki = 158.49 nM T21945 CDE7Z5 145978299 Ki = 5800 nM T21945 C87MSW 145980271 Ki = 458 nM T21945 CVKQ04 145981108 IC50 = 3710 nM T21945 CV1J4B 145981842 IC50 = 5130 nM T21945 C2A7WP 145982315 IC50 = 20500 nM T21945 CE0CB8 145983354 IC50 > 10000 nM T21945 CE84XH 145983742 IC50 > 10000 nM T21945 CO45RG 145983783 IC50 > 10000 nM T21945 C8F0IL 145983986 IC50 > 10000 nM T21945 CU53SY 145984002 IC50 > 10000 nM T21945 C9ZRP0 145984032 IC50 > 10000 nM T21945 CU6QS4 145984074 IC50 > 10000 nM T21945 CJ9UZ0 145984374 IC50 = 510 nM T21945 C6I3NT 145984803 IC50 > 10000 nM T21945 C7EIC6 145984821 IC50 > 10000 nM T21945 C6M1FI 145984939 IC50 = 3660 nM T21945 C9W6PO 145984940 IC50 > 10000 nM T21945 CT6KH5 145985061 IC50 = 260 nM T21945 CG2C8H 145985476 IC50 > 10000 nM T21945 C82KFY 145985630 IC50 = 23800 nM T21945 C1WA5L 145985747 IC50 = 1340 nM T21945 C1H2UT 145985812 IC50 > 10000 nM T21945 C5XC2O 145986024 IC50 = 3150 nM T21945 C5XCV8 145986058 IC50 = 2550 nM T21945 CG0Q1F 145986130 IC50 = 2690 nM T21945 CNJH37 145986752 Ki = 1438 nM T21945 CUGO10 145988693 Ki = 902 nM T21945 CW6E8Z 145989332 IC50 = 29700 nM T21945 C0X7BO 145990773 IC50 = 2540 nM T21945 CNBS32 145991101 IC50 = 5830 nM T21945 C5K3CS 145991656 IC50 = 2850 nM T21945 CBZY16 145993315 IC50 = 9740 nM T21945 CZP9L5 145993640 IC50 = 25900 nM T21945 CGTV18 145994198 IC50 = 1200 nM T21945 C6P3SR 153287553 Ki = 1584.89 nM T21945 CV9G7Z 153287572 Ki = 316.23 nM T21945 CO85KL 153287574 Ki = 398.11 nM T21945 C5LXC4 153605593 Ki = 4820 nM T21945 CDN5I4 155510548 IC50 = 67800 nM T21945 CYO17F 155510932 IC50 = 4000 nM T21945 C1Z7ED 155513346 IC50 = 10000 nM T21945 CH4Z9J 155513656 IC50 = 22700 nM T21945 CJ87WT 155514907 IC50 > 10000 nM T21945 CCF56N 155515030 IC50 = 230200 nM T21945 CF9PN2 155515352 IC50 = 365100 nM T21945 C5EQD6 155515957 IC50 = 1200 nM T21945 CB71XT 155517422 IC50 = 215500 nM T21945 CL0T5F 155517981 IC50 = 195800 nM T21945 CUSA24 155519891 Ki > 10000 nM T21945 CV5H7B 155521007 IC50 = 2050 nM T21945 CRM7H5 155521227 IC50 = 8870 nM T21945 CZLF49 155521764 IC50 = 4700 nM T21945 CWD38V 155524413 IC50 > 10000 nM T21945 CVF9H3 155524550 IC50 = 920 nM T21945 C8G6HD 155524923 IC50 = 1100 nM T21945 CVF9E8 155525067 IC50 = 68200 nM T21945 CX9PC3 155525160 IC50 = 89800 nM T21945 CHA8R7 155527331 IC50 = 38600 nM T21945 CFMJ93 155528557 IC50 = 261000 nM T21945 CJHX15 155529238 IC50 = 2160 nM T21945 CVNK03 155529810 IC50 = 36500 nM T21945 CC6X5O 155530123 IC50 = 350 nM T21945 CVLH72 155531187 IC50 = 73250 nM T21945 C2MB4H 155533557 IC50 = 1100 nM T21945 CC26GM 155534211 IC50 = 72000 nM T21945 CQV7D8 155534330 IC50 = 120800 nM T21945 CLTU63 155534741 IC50 = 164400 nM T21945 C0WX1T 155535629 IC50 > 10000 nM T21945 CB79ZW 155536080 Ki = 2511.89 nM T21945 CA25OD 155536376 IC50 = 85000 nM T21945 CRHA67 155536435 IC50 = 52560 nM T21945 CW37XJ 155543088 IC50 = 129300 nM T21945 C4STU5 155543525 Ki = 163 nM T21945 CB1F0Y 155545607 IC50 = 870 nM T21945 CE5YV0 155545747 IC50 > 10000 nM T21945 CI41YF 155546363 IC50 = 104300 nM T21945 CYOQ12 155546516 IC50 = 2480 nM T21945 C1URC8 155547273 Ki = 2109 nM T21945 CIK5C0 155547331 IC50 = 1060 nM T21945 CFW6O5 155547621 IC50 = 1450 nM T21945 CLH68U 155549829 IC50 > 10000 nM T21945 CAS6B5 155550042 Ki > 10000 nM T21945 CW0EG3 155550602 IC50 = 110500 nM T21945 C0UYA7 155551050 IC50 = 107300 nM T21945 CNG36O 155553448 IC50 = 1090 nM T21945 C1U2KX 155554780 IC50 > 10000 nM T21945 CH6ZD0 155556044 IC50 = 8540 nM T21945 CIU58J 155556193 IC50 = 163700 nM T21945 C6X2HA 155557651 IC50 = 1890 nM T21945 C8TO2W 155558029 Ki = 2800 nM T21945 CM5G9F 155558122 IC50 = 1720 nM T21945 C3E1DP 155558516 IC50 = 566400 nM T21945 CM0WK3 155558540 IC50 = 138800 nM T21945 C5B2OZ 155559232 Ki = 1082 nM T21945 C0I1YR 155559387 IC50 > 10000 nM T21945 CX1T3H 155559527 IC50 = 8200 nM T21945 C28MCV 155559835 Ki > 10000 nM T21945 C4O8LX 155560376 IC50 = 45490 nM T21945 C1FJ8G 155565910 IC50 = 107100 nM T21945 C6DQ1K 155566338 Ki = 5740 nM T21945 CN5P9D 155569039 IC50 = 109100 nM T21945 CVUR38 155569643 IC50 = 80 nM T21945 CP9TR0 10324985 Ki = 6980 nM T21945 CUKM52 44586281 Ki = 2770 nM T21945 CNG2T7 44586282 Ki = 6600 nM T21945 CP9ED8 44586283 Ki = 712 nM T21945 COY7T4 44586284 Ki = 1810 nM T21945 D00DEH 45483512 Ki = 13 nM T21945 D00FMX 46230706 Ki = 330 nM T21945 D00GDI 45487890 IC50 = 1670 nM T21945 D00HCC 12996705 Ki = 554 nM T21945 D00KRQ 23113096 Ki = 416 nM T21945 D00NEE 44413628 IC50 > 1000000 nM T21945 D00QCP 46837647 IC50 = 550 nM T21945 D00WMS 3047299 Ki = 5700 nM T21945 D01ABR 44414723 Ki = 31 nM T21945 D01AOI 44592200 IC50 = 1900 nM T21945 D01CXD 10398175 Ki > 10000 nM T21945 D01EIS 12263801 IC50 = 39 nM T21945 D01FFX 24691160 IC50 = 1800 nM T21945 D01GSG 44592199 IC50 = 772 nM T21945 D01JYY 11323940 IC50 = 1200 nM T21945 D01KAX 135453290 Ki > 10000 nM T21945 D01MBF 45483536 Ki = 97 nM T21945 D01RWY 44542656 IC50 = 2000 nM T21945 D01SHR 44593693 IC50 = 46 nM T21945 D01WWC 16573 Ki > 950 nM T21945 D01YED 45141808 IC50 = 718 nM T21945 D01YNZ 45483529 Ki = 76 nM T21945 D02DCM 44230874 Ki = 7 nM T21945 D02EKR 3031077 Ki > 10000 nM T21945 D02ENH 9797657 IC50 = 1995 nM T21945 D02ICX 14373 IC50 = 28.3 nM T21945 D02LQG 170832 Ki = 556 nM T21945 D02NUR 44543266 Ki > 10000 nM T21945 D02TMK 1614 IC50 = 266 nM T21945 D02YOO 4500 Ki = 1.6 nM T21945 D02YSN 11651575 IC50 = 2322 nM T21945 D02ZIQ 43227131 IC50 = 2520 nM T21945 D03BQV 3033806 IC50 = 40 nM T21945 D03DQQ 45375938 Ki = 18 nM T21945 D03EMO 16102754 IC50 = 49 nM T21945 D03FGM 44414732 IC50 > 400 nM T21945 D03HBZ 10850308 IC50 = 2100 nM T21945 D03HQF 11644566 IC50 = 59 nM T21945 D03JOX 11311147 IC50 = 19.7 nM T21945 D03MYV 44414735 IC50 = 73 nM T21945 D03YQY 46837650 IC50 = 1130 nM T21945 D03ZDY 44414750 IC50 = 35 nM T21945 D04KZX 44542809 IC50 = 135 nM T21945 D04NDO 45483400 Ki = 34 nM T21945 D04NKQ 22599992 Ki = 21 nM T21945 D04ZPF 45483409 Ki = 3 nM T21945 D05GDP 599482 Ki 10000 nM T21945 D05LJC 45483405 Ki = 9 nM T21945 D05LKO 44414722 Ki = 12 nM T21945 D05PLF 3031066 IC50 = 2070 nM T21945 D05UMA 10334821 IC50 = 13.2 nM T21945 D05ZUX 44207909 Ki >= 1000 nM T21945 D06CMJ 3127 IC50 = 207 nM T21945 D06EMC 11392888 Ki = 21 nM T21945 D06KNV 3703 Ki = 1.585 nM T21945 D06LCK 45141805 IC50 = 135 nM T21945 D06PJD 44593439 IC50 = 47 nM T21945 D06QGD 11357862 IC50 = 531 nM T21945 D06QIQ 44592241 IC50 = 4400 nM T21945 D06UDU 45483520 Ki = 115 nM T21945 D06WIV 44578367 Ki = 271 nM T21945 D07DWS 45483446 Ki = 526 nM T21945 D07IOX 44543268 Ki = 2580 nM T21945 D07LFR 44231007 Ki = 3 nM T21945 D07OOI 3456 IC50 = 165 nM T21945 D07PAT 16102753 IC50 = 180 nM T21945 D07SAA 44543271 IC50 = 2150 nM T21945 D07TEJ 44414874 IC50 > 400 nM T21945 D07ZOP 11470616 IC50 = 9.4 nM T21945 D08AWN 3058751 IC50 = 2806 nM T21945 D08EKQ 46890532 Ki = 30 nM T21945 D08JCK 16102777 IC50 = 220 nM T21945 D08JLB 45483406 Ki = 9 nM T21945 D08LAY 13904719 IC50 = 130 nM T21945 D08MEN 14014889 IC50 = 9100 nM T21945 D08NZE 126280 Ki = 15 nM T21945 D08RCH 44566054 IC50 > 10000 nM T21945 D08SCH 151900 IC50 = 2375 nM T21945 D08SLZ 16102764 Ki = 3.9 nM T21945 D09BYB 45487941 IC50 = 4100 nM T21945 D09DWM 44411213 Ki = 69 nM T21945 D09FIC 46890395 Ki = 28 nM T21945 D09HJL 10331436 Ki > 10000 nM T21945 D09IIH 45483459 EC50 = 358 nM T21945 D09JRN 44414721 IC50 = 300 nM T21945 D09QZM 11637187 IC50 = 58 nM T21945 D09RPR 16737207 Ki > 10000 nM T21945 D09VTJ 441298 IC50 = 2000 nM T21945 D09XWL 45141379 IC50 = 2850 nM T21945 D0A1HH 44414708 IC50 = 90 nM T21945 D0A3YK 44414860 IC50 > 400 nM T21945 D0A7GW 45487772 IC50 > 40000 nM T21945 D0AE9M 10801657 IC50 = 430 nM T21945 D0B4FN 11148955 IC50 = 56 nM T21945 D0B5AG 44560576 IC50 = 5000 nM T21945 D0BM0M 44454695 IC50 > 10000 nM T21945 D0BW0V 44589528 Ki = 89 nM T21945 D0C0GL 3031062 IC50 = 6500 nM T21945 D0C5GF 6918515 Ki > 10000 nM T21945 D0CG2Y 44133490 Ki = 2440 nM T21945 D0CK9K 6918513 Ki > 10000 nM T21945 D0D1KK 44410091 Ki = 148 nM T21945 D0D1RU 3081186 IC50 = 2500 nM T21945 D0D3QE 11550626 Ki > 10000 nM T21945 D0D5QV 9838803 IC50 = 6700 nM T21945 D0D8YY 44411431 Ki = 91 nM T21945 D0E3DM 44592118 IC50 = 2900 nM T21945 D0E6PQ 45483451 Ki = 170 nM T21945 D0EO5P 44414709 IC50 = 72 nM T21945 D0EX2M 44414720 IC50 = 54 nM T21945 D0F5AQ 49798218 Ki = 79.43 nM T21945 D0F5TA 10561859 IC50 = 250 nM T21945 D0F6GB 44133853 Ki = 74 nM T21945 D0FS4V 44413375 IC50 = 90000 nM T21945 D0G0CJ 45141380 IC50 = 2530 nM T21945 D0G1XP 44543273 IC50 = 43 nM T21945 D0G5RH 44462219 Ki = 550 nM T21945 D0G6BJ 24802842 Ki = 7.943 nM T21945 D0G8UA 46890321 Ki = 58 nM T21945 D0GG2J 46890492 Ki = 17 nM T21945 D0GY8R 45141807 IC50 = 577 nM T21945 D0H2TS 45483528 Ki = 1940 nM T21945 D0H4AD 44542509 IC50 = 2540 nM T21945 D0I2UC 44230733 Ki = 1 nM T21945 D0I4TO 10107888 IC50 = 445 nM T21945 D0I9KV 11220599 IC50 = 83 nM T21945 D0IB6Y 11658526 IC50 = 92 nM T21945 D0IC4J 45375937 Ki = 11 nM T21945 D0IR0R 16102751 IC50 = 50 nM T21945 D0J4CB 24803184 Ki = 10 nM T21945 D0J5AR 11672904 IC50 = 347 nM T21945 D0J5EF 215051 IC50 = 6500 nM T21945 D0J8DC 44414861 IC50 > 400 nM T21945 D0K3EW 49799108 Ki = 1 nM T21945 D0K6ZT 44133851 Ki = 536 nM T21945 D0KD9M 44592198 IC50 = 200 nM T21945 D0KS0I 24894910 Ki = 50 nM T21945 D0KT2M 44133674 Ki = 292 nM T21945 D0L0AY 11506691 IC50 = 360 nM T21945 D0L5MW 181743 Ki > 10000 nM T21945 D0L6RY 11322641 IC50 = 171 nM T21945 D0L7BK 44414856 IC50 = 48 nM T21945 D0M3TK 45483431 Ki = 1710 nM T21945 D0N0TQ 11571886 IC50 = 23 nM T21945 D0N2KU 44517677 Ki = 6 nM T21945 D0N2RJ 45483432 Ki = 1720 nM T21945 D0NC3P 117443 IC50 > 200000 nM T21945 D0NM1F 45487774 IC50 = 7500 nM T21945 D0NY4W 11152502 IC50 = 46.5 nM T21945 D0O2LC 44543272 IC50 > 100 nM T21945 D0O9BL 11210506 IC50 = 81 nM T21945 D0P6SY 14595987 IC50 = 880 nM T21945 D0P8BE 10635415 IC50 = 1300 nM T21945 D0P9EO 45141381 IC50 = 8700 nM T21945 D0Q6SH 45483408 Ki = 170 nM T21945 D0Q8IQ 43794735 IC50 = 1520 nM T21945 D0R1AE 44332186 Ki = 46700 nM T21945 D0R1XT 10799123 IC50 = 1000 nM T21945 D0R3TA 45483407 Ki = 162 nM T21945 D0R5AD 43227726 Ki = 4476 nM T21945 D0R8EV 3027752 IC50 = 969 nM T21945 D0R8TH 16102750 IC50 = 210 nM T21945 D0RT9B 11506733 IC50 = 61 nM T21945 D0S1XC 25224941 IC50 = 9 nM T21945 D0S4JT 45483466 Ki = 183 nM T21945 D0S9AY 44592244 IC50 = 10500 nM T21945 D0S9IO 44454825 IC50 = 450 nM T21945 D0SN6R 44592197 IC50 = 1400 nM T21945 D0T2RY 9948320 Ki >= 1000 nM T21945 D0T5VG 11514389 IC50 = 3420 nM T21945 D0T8BU 13904714 IC50 = 14 nM T21945 D0U3SB 45141806 IC50 = 1180 nM T21945 D0U7OD 16043230 Ki = 12 nM T21945 D0V0PR 45483527 Ki = 1710 nM T21945 D0V4FW 24861406 Ki = 792 nM T21945 D0V5GB 11637190 Ki = 58.88 nM T21945 D0V8IZ 44543267 IC50 = 400 nM T21945 D0V9SV 44559130 IC50 = 6040 nM T21945 D0VC1K 826600 IC50 = 70 nM T21945 D0VY9K 45141809 IC50 = 4100 nM T21945 D0W5IN 10515839 IC50 = 1100 nM T21945 D0W6WL 44414840 IC50 > 400 nM T21945 D0W8BJ 44560674 IC50 = 840 nM T21945 D0W8YO 46230654 EC50 = 28 nM T21945 D0W9JK 11220185 IC50 = 24 nM T21945 D0WB6P 46227262 IC50 = 188 nM T21945 D0X3CF 442879 IC50 = 8760 nM T21945 D0X8GC 45487773 IC50 > 40000 nM T21945 D0X8LG 11243002 IC50 = 11.7 nM T21945 D0XF5P 44592119 IC50 = 1200 nM T21945 D0XY9E 3029724 IC50 = 370 nM T21945 D0Y1MJ 16102749 IC50 = 35 nM T21945 D0Y3BI 11572135 IC50 = 210 nM T21945 D0Y5CG 45483467 Ki = 104 nM T21945 D0Y6GQ 44414862 IC50 > 400 nM T21945 D0Y7CS 44543118 IC50 = 6200 nM T21945 D0Y8UC 3929516 Ki = 844 nM T21945 D0Z4UF 10524711 IC50 = 750 nM T21945 D0Z5GR 46230818 Ki = 747 nM T21945 D0Z6YA 11289879 IC50 = 16 nM T21945 D0Z9OX 44414719 IC50 = 22 nM T21945 D0ZC3Q 44230732 Ki = 1 nM T21945 D0ZE4C 45141608 IC50 = 8200 nM T21945 D0ZS3M 10490725 IC50 = 680 nM T21945 D0ZU5W 22615724 EC50 = 83 nM T81637 D05MQK 110635 IC50 > 10000 nM T81637 D0Z7ZM 135398744 IC50 = 600 nM T81637 D01LCC 17754438 IC50 > 10000 nM T81637 D0SM0W 44591583 IC50 = 6100 nM T81637 D0T5PO 5092 IC50 > 50000 nM T81637 D05VBJ 71295299 IC50 > 10000 nM T81637 C0YK8A 155806 IC50 = 10000 nM T81637 CIR61A 188375 IC50 = 350 nM T81637 CF62QN 275182 IC50 = 22000 nM T81637 C1B6ZL 662965 IC50 > 50000 nM T81637 CZH08Y 9802738 IC50 > 20000 nM T81637 C1B4XD 11992634 IC50 > 2000 nM T81637 CPX16N 11993169 IC50 > 2000 nM T81637 C20VHK 24871823 IC50 = 580 nM T81637 C6EQG2 24963293 IC50 > 2000 nM T81637 CQU19I 44180409 IC50 = 118 nM T81637 CW8OB3 44243146 Ki > 10000 nM T81637 C5IMB2 46239424 Ki > 10000 nM T81637 CKR9P7 46239425 Ki > 10000 nM T81637 C3P2IN 46933992 IC50 >= 58000 nM T81637 CPC3T4 56654131 IC50 > 10000 nM T81637 CD52CA 57391118 IC50 > 2000 nM T81637 CG3DF1 57392948 Ki > 10000 nM T81637 CE36TV 57394695 Ki > 10000 nM T81637 CPA3D1 57403394 Ki > 10000 nM T81637 CWX3N7 59320301 IC50 = 462 nM T81637 C0EP5I 59341847 IC50 > 10000 nM T81637 CHQ28A 59341978 IC50 > 10000 nM T81637 C4P0XT 71092344 IC50 = 7400 nM T81637 C6DAG4 71092519 IC50 = 25600 nM T81637 C2HGI7 71153408 IC50 > 10000 nM T81637 C7XRY6 72190879 IC50 = 2497 nM T81637 CBM61I 73293715 IC50 = 452 nM T81637 C9JE6M 75815419 IC50 = 42 nM T81637 CSCY01 117949009 IC50 = 2000 nM T81637 CRJE23 122185011 IC50 = 2 nM T81637 CS6M9C 122193679 IC50 > 100000 nM T81637 C2P1IU 134129996 IC50 > 100000 nM T81637 CLE03O 134130328 IC50 > 100000 nM T81637 CSN6J0 134130563 IC50 > 100000 nM T81637 C0A1CZ 134131162 IC50 > 100000 nM T81637 CZ09EG 135418212 IC50 = 54 nM T81637 C7GC0D 135436665 IC50 > 10000 nM T81637 C3R8SE 135457869 IC50 = 3900 nM T81637 CWQG94 135484473 IC50 = 2500 nM T81637 CX7I5Z 135721222 IC50 = 1430 nM T81637 CTX54Z 135896326 IC50 = 7700 nM T81637 CH6QL0 136059722 IC50 = 790 nM T81637 C2J7ZU 136059723 IC50 > 10000 nM T81637 CN06GO 136059724 IC50 > 10000 nM T81637 C8EA6G 136059725 IC50 > 10000 nM T81637 C31KAG 136059726 IC50 > 10000 nM T81637 C12UMG 136059728 IC50 > 10000 nM T81637 C21FVA 136180322 IC50 = 62 nM T81637 C2N9VT 137348687 IC50 > 10000 nM T81637 C2QLX3 138393292 IC50 > 50000 nM T81637 CSOF52 141737655 IC50 > 20000 nM T81637 C7SRA2 141737657 IC50 > 20000 nM T81637 CMIY07 141737666 IC50 > 20000 nM T81637 CC61SD 141737667 IC50 > 20000 nM T81637 C14CZJ 141737668 IC50 > 20000 nM T81637 CTNG49 141737674 IC50 > 20000 nM T81637 CJ38IC 141737676 IC50 > 20000 nM T81637 C1MC5Z 141737681 IC50 > 20000 nM T81637 CTUL23 141737690 IC50 > 20000 nM T81637 CMW20N 141737696 IC50 > 20000 nM T81637 CO1C4S 141737703 IC50 > 20000 nM T81637 CX9N1P 141737704 IC50 > 20000 nM T81637 C8HEG7 141737705 IC50 > 20000 nM T81637 C4W2YJ 145961173 IC50 = 777 nM T81637 CC7HN2 145974174 IC50 > 100000 nM T81637 CK1BR0 145978345 IC50 > 100000 nM T81637 CL8CU6 155521936 IC50 > 200000 nM T81637 CT85RG 155530589 IC50 > 200000 nM T81637 D09RKU 46239428 Ki > 10000 nM T54982 CR9E3G 690945 IC50 = 1480 nM T54982 CD5HM0 774146 IC50 = 160 nM T54982 C93YWR 1105962 IC50 = 3440 nM T54982 C9KEX6 1292961 IC50 > 10000 nM T54982 C7ZI4W 2169492 IC50 = 280 nM T54982 COT0J8 2352151 IC50 = 1950 nM T54982 C3C7SM 4815751 IC50 = 6010 nM T54982 CJ0X3Q 9243420 IC50 = 270 nM T54982 CPO58R 15950502 IC50 = 260 nM T54982 C2TOM4 15950504 IC50 = 477 nM T54982 CV30SC 15950714 IC50 = 34 nM T54982 CIGO41 15950719 IC50 = 36 nM T54982 C2JWD0 15950720 IC50 = 71 nM T54982 COF3W0 15950791 IC50 = 77 nM T54982 CP84DN 15950792 IC50 = 270 nM T54982 C13YRK 15950862 IC50 = 7080 nM T54982 CG83IP 15950863 IC50 = 1300 nM T54982 CFE89M 15950864 IC50 = 230 nM T54982 CN4XI2 15950866 IC50 = 190 nM T54982 CSV95U 15950936 IC50 = 1260 nM T54982 CF4Z3T 15950992 IC50 = 21 nM T54982 CU4QW5 15951121 IC50 = 76 nM T54982 C3YBA6 15951123 IC50 = 52 nM T54982 C78WBD 15951124 IC50 = 653 nM T54982 C6XU0R 15951185 IC50 = 2180 nM T54982 CF9XO7 15951399 IC50 = 73 nM T54982 CXPJ41 15951403 IC50 = 146 nM T54982 CW2J4G 15951469 IC50 = 190 nM T54982 C9GA4T 17427022 IC50 = 7010 nM T54982 CQ3VP7 24539421 IC50 = 2230 nM T54982 CKU1J3 26519893 IC50 = 2700 nM T54982 CC9KS4 31532942 IC50 > 10000 nM T54982 CI09TN 58754889 IC50 = 36 nM T54982 CK74ZO 68700057 IC50 = 5000 nM T54982 C0SVP5 110756102 IC50 = 1880 nM T54982 C8YBH1 118708988 IC50 = 150 nM T54982 CNO51X 118708989 IC50 = 34 nM T54982 CCK1Z5 118708990 IC50 = 61 nM T54982 CY0FE3 118708991 IC50 = 1020 nM T54982 CM17XS 118708992 IC50 = 870 nM T54982 C43RPJ 118708993 IC50 > 10000 nM T54982 CG60XU 118708994 IC50 > 10000 nM T54982 CV0ZH2 118708995 IC50 = 700 nM T54982 CP4CS3 118708996 IC50 = 53 nM T54982 CK68MY 118708997 IC50 = 24 nM T54982 COTP85 118708998 IC50 = 76 nM T54982 CMJ9L6 118708999 IC50 = 128 nM T54982 CKSO64 118709000 IC50 = 392 nM T54982 CBQ63T 118709001 IC50 = 57 nM T54982 C1CDG6 118709002 IC50 = 89 nM T54982 CSCD98 118709003 IC50 = 586 nM T54982 CS74UO 118709004 IC50 = 1340 nM T54982 CQU5P7 118709005 IC50 = 27 nM T54982 D0M6UK 91827366 IC50 = 18 nM T13491 D06IAR 60961 Ki = 12000 nM T13491 D0F9GE 3108 Ki = 8.18 nM T13491 D0L7VL 3926 Ki = 279.9 nM T13491 D0Y7DP 6029 Ki = 51000 nM T13491 D00YSJ 158795 Ki = 11000 nM T13491 CHU7Q8 9570 IC50 = 229086.77 nM T13491 CX0YR8 20345 IC50 = 36307.81 nM T13491 CCL04N 65519 IC50 = 66.1 nM T13491 CS4QG5 92208 IC50 = 10715.19 nM T13491 CP23YX 95846 IC50 = 57543.99 nM T13491 C5Q7PG 97297 IC50 = 229086.77 nM T13491 CYH2X7 97481 IC50 = 27.54 nM T13491 C7V2ON 101430 IC50 = 32359.37 nM T13491 CQJ96I 125347 IC50 = 4168.69 nM T13491 CQY72X 162449 IC50 = 2.754 nM T13491 C63QWR 171030 Ki = 14.23 nM T13491 CCD16T 234001 IC50 = 275422.87 nM T13491 CUG20L 237307 IC50 = 218776.16 nM T13491 COQ7T4 240888 IC50 = 144543.98 nM T13491 C1D0QI 240890 IC50 = 120226.44 nM T13491 CSPI94 241405 IC50 = 63095.73 nM T13491 CRS4Y7 242656 IC50 = 91201.08 nM T13491 CQR46O 242658 IC50 = 52480.75 nM T13491 CQ40MW 350854 Ki = 393 nM T13491 CK05YL 350886 Ki = 216.4 nM T13491 CX0IF1 350887 Ki = 216.7 nM T13491 C63ZWC 408168 IC50 = 234422.88 nM T13491 C43HPC 408176 IC50 = 100000 nM T13491 CY8TR6 3006525 IC50 = 389045.14 nM T13491 C58HXO 3009565 Ki = 67.61 nM T13491 C03HUS 3009566 Ki = 99.49 nM T13491 C8A9IP 3009567 Ki = 16.22 nM T13491 C0CU6A 3009568 Ki = 19.05 nM T13491 CUB05H 3009569 Ki = 1.778 nM T13491 C7EA1J 3009570 Ki = 15.14 nM T13491 C3UEZ8 3009571 Ki = 7.079 nM T13491 CM0T4C 3009572 Ki = 9.98 nM T13491 C0YK9H 3009573 Ki = 34.67 nM T13491 C6TUM2 3009574 Ki = 10000 nM T13491 C9W1LK 3009575 Ki = 46.77 nM T13491 C4VBC9 3009576 Ki = 4.571 nM T13491 CBD20N 3009577 Ki = 9.02 nM T13491 C0HC7Q 3009578 Ki = 4.365 nM T13491 CW31PT 3009579 Ki = 87.1 nM T13491 CIR9H0 3009580 Ki = 12.59 nM T13491 CA9N7U 3010379 IC50 = 194984.46 nM T13491 CHU18X 3010380 IC50 = 338844.16 nM T13491 C4P1LX 3010387 IC50 = 114815.36 nM T13491 C4RK8O 3010388 IC50 = 77624.71 nM T13491 CIQN05 6477178 Ki = 19.95 nM T13491 CF4SL6 6480503 Ki = 19.87 nM T13491 C47RCN 6480761 Ki = 1905.46 nM T13491 CDI5A7 9850791 Ki = 91.6 nM T13491 C9LCJ7 9910431 Ki = 0.45 nM T13491 CI5Y2P 10046039 Ki = 97 nM T13491 CH1N3P 10098211 Ki = 39 nM T13491 C5UBA4 10150952 Ki = 1637 nM T13491 CB58VE 10255410 Ki = 3.802 nM T13491 CP4O2E 10287739 Ki = 4877 nM T13491 C08CYB 10340530 Ki = 39 nM T13491 C04XVO 10407876 IC50 = 114815.36 nM T13491 C9QI0R 10993654 Ki = 250 nM T13491 CY20OX 10993655 Ki = 300 nM T13491 C53SFO 11003496 Ki = 150 nM T13491 C8ERU0 11004466 Ki = 15 nM T13491 CRJ4X9 11165273 Ki = 124 nM T13491 CK31OX 11165691 Ki = 110 nM T13491 CNG96Y 11165692 Ki = 264 nM T13491 CX7JB3 11166106 Ki = 200 nM T13491 CF87NE 11167057 Ki = 129 nM T13491 CZ5SL1 11167331 Ki = 93 nM T13491 CXI51R 11176386 Ki = 2709 nM T13491 C2E6HZ 11188925 Ki = 488 nM T13491 CGI9X1 11201689 Ki = 1519 nM T13491 CR72AQ 11212078 Ki = 212 nM T13491 C1EI5Y 11259978 Ki = 111 nM T13491 CWM91U 11272406 Ki = 86 nM T13491 C05YXB 11292364 Ki = 3340 nM T13491 C3T4CJ 11294339 Ki = 196 nM T13491 C7LU3C 11302153 IC50 = 13489.63 nM T13491 CFZQ07 11303957 Ki = 153 nM T13491 CH7BV4 11350617 Ki = 325.2 nM T13491 C9FCH3 11351695 Ki = 51 nM T13491 CZV6W2 11361323 Ki = 711 nM T13491 CQE09C 11363502 Ki = 55 nM T13491 CXZ14N 11397549 Ki = 225 nM T13491 CMLG74 11397550 Ki = 221 nM T13491 CQ8C5A 11429692 Ki = 563 nM T13491 C78GYL 11453959 Ki = 29 nM T13491 C4LU6P 11454136 Ki = 126 nM T13491 CXF8T6 11464060 Ki = 236 nM T13491 C6NR2G 11465833 Ki = 104 nM T13491 CN5YJ7 11474405 Ki = 2165 nM T13491 CSL34W 11476919 Ki = 154 nM T13491 CCL7X8 11477414 Ki = 422 nM T13491 CN85OM 11751510 Ki = 89 nM T13491 C5QVZ1 11775148 Ki = 2165 nM T13491 CVOA06 11784658 Ki = 196 nM T13491 CBU15I 11796049 IC50 = 181.97 nM T13491 C5HJ2Z 12298620 Ki = 690.9 nM T13491 C9L4US 13506394 IC50 = 257039.58 nM T13491 CSXT86 14544367 IC50 = 575439.94 nM T13491 CE1W0F 15728777 IC50 = 93.9 nM T13491 C3VJH5 16755878 Ki = 38 nM T13491 CVS39W 16755880 Ki = 16.8 nM T13491 C5LZ4M 16755882 Ki = 139.9 nM T13491 C1XLE8 16755977 Ki = 120.7 nM T13491 CAQV24 16755979 Ki = 14.7 nM T13491 C8P1EA 16755981 Ki = 427.6 nM T13491 CNO78X 16756082 Ki = 104.1 nM T13491 CNL27G 16756084 Ki = 15.8 nM T13491 C1IEU7 16756086 Ki = 53.1 nM T13491 C1HE0Q 16756299 Ki = 4.3 nM T13491 C5E4RI 16756300 Ki = 99.7 nM T13491 CL7JD4 16756414 Ki = 0.86 nM T13491 CX8OT1 16756415 Ki = 0.49 nM T13491 CV38RS 16756416 Ki = 38 nM T13491 CW81NT 16757073 Ki = 449 nM T13491 C7V6LI 16757076 Ki = 21.2 nM T13491 CT1X8Q 16757077 Ki = 0.77 nM T13491 C8CT7W 16757477 Ki = 300 nM T13491 CJ4M8V 16757479 Ki = 191 nM T13491 C6PEN2 16757481 Ki = 136 nM T13491 C32PNB 16757482 Ki = 489 nM T13491 C8BAI3 17860366 Ki = 361 nM T13491 CVB8G5 17860373 Ki = 130 nM T13491 CDA87V 17860381 Ki = 1544 nM T13491 CFQ0K4 17860382 Ki = 281 nM T13491 CM3B9O 17860386 Ki = 653 nM T13491 C5NG4X 20055595 IC50 = 33.11 nM T13491 CN0A3O 21139659 IC50 = 13803.84 nM T13491 C9FXD0 21139665 IC50 = 13489.63 nM T13491 CR0X3M 21139723 IC50 = 2884.03 nM T13491 CI46ZU 21144233 IC50 = 63095.73 nM T13491 C2GY7O 21820756 IC50 = 204173.79 nM T13491 CVI2K0 24809875 Ki = 2.1 nM T13491 CQ52MX 24860453 Ki = 193 nM T13491 CV7P6G 24860459 Ki = 8.2 nM T13491 CWT4Z5 24860460 Ki = 17.1 nM T13491 C0ZS5G 24894638 IC50 = 5248.07 nM T13491 C4GHC8 25195323 Ki > 1000000 nM T13491 CCA6B2 44437757 Ki = 24 nM T13491 COPC72 44437758 Ki = 429 nM T13491 CGZ3W7 44437759 Ki = 24 nM T13491 CSA9R5 44437760 Ki = 193 nM T13491 C14JTW 44437761 Ki = 25 nM T13491 CW81EM 44437762 Ki = 325 nM T13491 C6CFP7 44437763 Ki = 33 nM T13491 CC2AP9 44437764 Ki = 357 nM T13491 CNE01K 44437765 Ki = 125 nM T13491 COX2B7 44437766 Ki = 400 nM T13491 C3IEQ8 44437767 Ki = 247 nM T13491 CBRA57 44437768 Ki = 394 nM T13491 CDC7S3 44437769 Ki = 86 nM T13491 CB5G9Y 44437770 Ki = 243 nM T13491 C1G4ZI 44437771 Ki = 11 nM T13491 C2UBD4 44437772 Ki = 11 nM T13491 CW6I1S 44437773 Ki = 11 nM T13491 COW9H0 44437775 Ki = 34 nM T13491 CR5Q6C 44437776 Ki = 315 nM T13491 CY45AO 44450834 IC50 = 223.87 nM T13491 CC6NT7 44450837 IC50 = 812.83 nM T13491 CHCF10 44450839 Ki = 18.89 nM T13491 C0LVG1 44450840 Ki > 1000 nM T13491 CXVF19 44450855 IC50 = 707.95 nM T13491 CZ6OS3 44450858 IC50 = 281.84 nM T13491 CLN3P8 44450861 IC50 = 354.81 nM T13491 CGB3S4 44450863 IC50 = 5248.07 nM T13491 CA45IY 44450864 Ki > 1000 nM T13491 CPXD89 44450865 Ki > 1000 nM T13491 C4L9VM 44450880 IC50 = 1174.9 nM T13491 C7U3OZ 44450883 IC50 = 977.24 nM T13491 CSIY54 44450884 IC50 = 1778.28 nM T13491 CSU7Z1 44450885 IC50 = 87.1 nM T13491 CNY01F 44450887 IC50 = 1513.56 nM T13491 C3RT0Z 44450910 IC50 = 2398.83 nM T13491 C15ATB 44450911 IC50 = 1288.25 nM T13491 C3FY9P 44450912 IC50 = 33113.11 nM T13491 C2E4QH 44450913 IC50 = 77.62 nM T13491 C6O2TY 44450939 IC50 = 46773.51 nM T13491 C0KJ4H 44450940 IC50 = 15.85 nM T13491 C4AV6K 44450946 IC50 = 91201.08 nM T13491 CJZR25 44450962 IC50 = 346.74 nM T13491 CD7IL5 44450963 IC50 = 426.58 nM T13491 CGPE70 44450987 IC50 = 31.62 nM T13491 C7QCF0 44451028 IC50 = 616.6 nM T13491 C3K4QX 44451029 IC50 = 331131.12 nM T13491 CIU31R 44451031 IC50 = 123.03 nM T13491 C7A0YM 44451032 IC50 = 14454.4 nM T13491 C70YLH 44451034 IC50 = 1348.96 nM T13491 C5-MAY-03 44451035 IC50 = 446683.59 nM T13491 CQNZ28 44451058 IC50 = 14791.08 nM T13491 CFV3Q6 44451059 IC50 = 69.18 nM T13491 CH3G2N 44451060 IC50 = 34673.69 nM T13491 CJ2CV8 44451061 IC50 = 32359.37 nM T13491 C6GEV7 44451062 IC50 = 114815.36 nM T13491 C2MGW8 44451063 IC50 = 4786.3 nM T13491 C8GSW2 44451082 IC50 = 158.49 nM T13491 C1LUC4 44451083 IC50 = 251.19 nM T13491 CXJO71 44451084 IC50 = 16218.1 nM T13491 CS60YL 44451086 IC50 = 177.83 nM T13491 C8ITL7 44451087 IC50 = 21379.62 nM T13491 COJ08L 44451088 IC50 = 1548.82 nM T13491 CTW61X 44451089 IC50 = 6309.57 nM T13491 CA4TY1 44451113 IC50 = 812.83 nM T13491 CNM28K 44451114 IC50 = 81.28 nM T13491 C57DFP 44451115 IC50 = 4570.88 nM T13491 CP4YT5 44451116 IC50 = 11481536.21 nM T13491 CTJV12 44451136 IC50 = 21.88 nM T13491 CEO29K 44451137 IC50 = 177.83 nM T13491 CS08IW 44451139 IC50 = 4.786 nM T13491 C8N1WU 44451141 IC50 = 41686.94 nM T13491 CGU41Z 44451142 IC50 = 2089.3 nM T13491 CX34EG 44451143 IC50 = 190546.07 nM T13491 CQT8F6 44451144 IC50 = 17782.79 nM T13491 C4U5JC 44451174 IC50 = 107.15 nM T13491 CB83NF 44451176 IC50 = 245.47 nM T13491 C3T8FH 44451177 IC50 = 199.53 nM T13491 CFJ1H7 44451178 IC50 = 81283.05 nM T13491 CVMS06 44451179 IC50 = 8709.64 nM T13491 CWY34O 44451180 IC50 = 309.03 nM T13491 C93HJN 44451204 IC50 = 331.13 nM T13491 CO15ZC 44451205 IC50 = 281.84 nM T13491 C56MPX 44451207 IC50 = 1148.15 nM T13491 CBM85Q 44451208 IC50 = 162181.01 nM T13491 CI8JD3 44451209 IC50 = 4786.3 nM T13491 CBE50D 44451213 IC50 = 912010.84 nM T13491 C35AYJ 44451234 IC50 = 363.08 nM T13491 C1MZQ2 44451235 IC50 = 12022.64 nM T13491 CFYI73 44591161 Ki = 11.21 nM T13491 CB5O2L 44591162 Ki = 15.96 nM T13491 C85XLY 44591189 Ki = 134.23 nM T13491 CL9Z1G 44591190 Ki = 20.54 nM T13491 CQK0S2 44591191 Ki = 16.13 nM T13491 C40XZE 44591192 Ki = 13.79 nM T13491 C1J4QG 44591237 Ki = 38.9 nM T13491 CQ7NU4 44591238 Ki = 36.31 nM T13491 CU2OM7 44591239 Ki = 114.82 nM T13491 CBIH37 45487313 Ki = 0.064 nM T13491 CC53EM 45487314 Ki = 0.018 nM T13491 CXJA28 46877070 Ki = 5.4 nM T13491 C1OQK4 46877071 Ki = 0.94 nM T13491 CZYH80 46877077 Ki = 744 nM T13491 CME56L 46877100 Ki = 3 nM T13491 C48GIS 46877135 Ki = 0.64 nM T13491 C13KTE 46877136 Ki = 3.7 nM T13491 CPDI81 46877137 Ki = 3.6 nM T13491 CN25GX 46877164 Ki = 410 nM T13491 CO58LR 46877165 Ki = 9.5 nM T13491 C57WNU 46877166 Ki = 5.3 nM T13491 CG79UC 46877168 Ki = 28 nM T13491 C1EV5U 46877189 Ki = 2.3 nM T13491 CDG84T 50896860 IC50 = 4.6 nM T13491 CL4FI8 50896883 IC50 = 217 nM T13491 C97IFC 50896884 IC50 = 2.8 nM T13491 CK26LG 50944048 IC50 = 803 nM T13491 CBPQ23 56589406 IC50 = 31 nM T13491 C3U0ND 56589419 IC50 = 17.7 nM T13491 C9SZU7 76369267 IC50 = 3.2 nM T13491 D00GUM 3074 IC50 = 17.5 nM T13491 D02TOP 65407 IC50 = 0.3 nM T13491 D03RFA 657378 Ki = 1100 nM T13491 D06WAL 6072 Ki > 1000000 nM T13491 D09FHE 96048 Ki = 1.1 nM T13491 D0I7ON 10237315 Ki = 135 nM T13491 D0V8DJ 11165248 Ki = 2200 nM T02591 C26SVD 451777 IC50 = 250000 nM T02591 C5ZJQ3 488950 IC50 = 30000 nM T02591 C7GFT4 488962 IC50 > 100000 nM T02591 C8Q9JO 16134139 IC50 = 0.86 nM T02591 C7EC9G 16134140 IC50 = 0.84 nM T02591 C3A0YM 16134186 IC50 = 0.34 nM T02591 C6JQ3C 16143364 IC50 = 0.35 nM T02591 C6PG2R 46186917 IC50 = 9600 nM T02591 C9HL2I 46200686 IC50 = 9300 nM T02591 CRC8H5 53324414 IC50 = 83200 nM T02591 CG64CF 71596849 IC50 = 2.18 nM T02591 CZ7R4M 71597777 IC50 = 2.27 nM T02591 C8ML9U 122184656 IC50 = 17.74 nM T02591 C0FJ8S 122184657 IC50 = 17.7 nM T02591 CZ1R0G 122184658 IC50 > 2250 nM T02591 CF5P4J 122184659 IC50 = 58.79 nM T02591 D03QJA 11718722 IC50 = 1.71 nM T09528 D0NR6S 3002977 IC50 = 0.0024 ug.mL-1 T09528 CG5EA4 46222002 IC50 > 100 ug.mL-1 T09528 CH96GT 46871630 IC50 = 22.64 ug.mL-1 T09528 C3G7BP 71450125 IC50 = 28.6 ug.mL-1 T09528 CTE2J1 71450127 IC50 = 5.9 ug.mL-1 T09528 CVS14E 71453764 IC50 > 100 ug.mL-1 T09528 CV9I6A 71453766 IC50 = 80.92 ug.mL-1 T09528 CUJ52B 71457283 IC50 = 10.25 ug.mL-1 T09528 C6ENV5 100951623 EC50 > 10000 nM T00884 D09GOS 2812 IC50 = 7900 nM T00884 D0K8KX 5280343 IC50 = 4500 nM T00884 D0TG1H 3033 IC50 = 12 nM T00884 D00QKI 9865554 IC50 = 3.9 nM T00884 D00XBC 46861584 IC50 > 10000 nM T00884 D0LJ1B 9838712 IC50 = 1 nM T00884 D0O2XQ 11256587 IC50 > 10000 nM T00884 D0SN7I 10479502 IC50 > 10000 nM T00884 D0F6WV 3854666 IC50 = 22 nM T00884 CY4WG9 3793 IC50 = 5011.87 nM T00884 C3VL8J 9836859 IC50 = 6700 nM T00884 CVQ8J1 9843640 IC50 = 2000 nM T00884 CAN73G 9868309 IC50 = 4317 nM T00884 CCI9Y7 9888410 IC50 = 1366 nM T00884 C5C7OU 9912703 IC50 = 55 nM T00884 CEC1R6 9951571 IC50 = 13360 nM T00884 CYZT87 9953415 IC50 = 2600 nM T00884 C91RTG 9956238 IC50 > 10000 nM T00884 CNAI53 9968028 IC50 = 910 nM T00884 CLA2Z1 9968185 IC50 = 7600 nM T00884 C4MJ6R 9978981 Ki = 50 nM T00884 CE58ON 10027494 Ki = 283 nM T00884 CO37XS 10112327 IC50 = 2100 nM T00884 CR0ZQ6 10127252 Ki = 6 nM T00884 CP31MV 10150526 IC50 = 26 nM T00884 CG86FS 10150721 Ki = 9 nM T00884 C4SBE6 10157580 IC50 = 10500 nM T00884 C6VTZ4 10158569 IC50 = 9600 nM T00884 CRD2Z1 10180509 Ki = 123 nM T00884 CTU8G7 10194831 Ki = 6 nM T00884 CG2F7V 10200589 Ki = 40 nM T00884 CR6X8O 10201676 IC50 = 197 nM T00884 C59YEV 10224934 Ki = 21 nM T00884 CK14RC 10225736 Ki = 41 nM T00884 CD50IY 10237849 Ki = 7 nM T00884 C0C1GZ 10238257 Ki = 9 nM T00884 CXV73N 10252538 Ki = 10 nM T00884 C4L2TP 10252630 Ki = 11 nM T00884 CK49NQ 10272003 IC50 > 10000 nM T00884 C96NCK 10272255 IC50 = 81 nM T00884 C5HB3J 10291817 IC50 = 3900 nM T00884 CTH2M9 10292991 IC50 = 3000 nM T00884 C1U2KT 10293321 IC50 = 67 nM T00884 CR17PX 10294353 IC50 = 179 nM T00884 CR3PW7 10295195 IC50 = 2500 nM T00884 CL0K5B 10298837 IC50 = 22700 nM T00884 CKHY86 10310100 Ki = 3 nM T00884 CTWQ06 10343142 Ki = 10 nM T00884 CL4G6W 10389383 IC50 = 230 nM T00884 CF9T6H 10411524 Ki = 53 nM T00884 C2CAD9 10412163 Ki = 16 nM T00884 C8LIQ4 10478354 Ki = 34 nM T00884 C3R7XL 10481927 Ki = 14 nM T00884 C68OUD 10555185 IC50 = 5500 nM T00884 C1DYJ3 10578242 IC50 = 20000 nM T00884 CI2SN0 11222420 IC50 = 12000 nM T00884 CA39QR 11227406 IC50 > 10000 nM T00884 C20CDG 11245544 IC50 = 4200 nM T00884 CQ6KW0 11272103 IC50 = 10000 nM T00884 CJS9C0 11304851 IC50 = 7600 nM T00884 C1A5ET 11329244 IC50 = 10000 nM T00884 CL24DX 11371755 IC50 = 24000 nM T00884 CA1NU5 11750288 IC50 = 3200 nM T00884 CH3BX2 11798740 IC50 = 4500 nM T00884 C5X7MU 16098480 IC50 = 145 nM T00884 CQGO53 16098481 IC50 = 775 nM T00884 CR4AX9 16098482 IC50 = 34 nM T00884 CFX6N0 16098485 IC50 = 3058 nM T00884 C1BXN5 16098486 Ki = 146 nM T00884 CH2S4D 16098487 IC50 = 55 nM T00884 CUPD35 16098488 IC50 = 11 nM T00884 CEF6N1 16126703 IC50 = 6204 nM T00884 CQ2V9Y 21037713 IC50 = 99 nM T00884 CPJ3A2 21184843 IC50 = 11100 nM T00884 CGM3N9 23709380 IC50 = 0.1 nM T00884 CJ9E8V 25110787 IC50 = 917 nM T00884 C0PIM7 42642630 Ki = 6 nM T00884 CKQ82X 44157035 Ki = 8 nM T00884 C1LCP6 44249825 Ki = 381 nM T00884 CJ5CR2 44393537 IC50 = 4400 nM T00884 CU9K6S 44393538 IC50 = 5400 nM T00884 C1GB4Z 44393540 IC50 = 10600 nM T00884 CF64GM 44393541 IC50 = 6037 nM T00884 CGJE30 44393543 IC50 = 30000 nM T00884 C0VL5O 44393568 IC50 = 12100 nM T00884 CH91YQ 44393569 IC50 = 8100 nM T00884 CRI97S 44393573 IC50 < 30000 nM T00884 CE09WT 44393592 IC50 = 2700 nM T00884 CRNZ65 44393593 IC50 = 3100 nM T00884 C8HP1A 44393655 IC50 = 1600 nM T00884 CN10IS 44393659 IC50 = 8900 nM T00884 COS64B 44393699 IC50 = 6200 nM T00884 C9M2HX 44393730 IC50 = 11500 nM T00884 C8SE3I 44393748 IC50 = 6000 nM T00884 CI74SU 44393777 IC50 > 25000 nM T00884 CCMI24 44419411 IC50 = 512 nM T00884 C39AZS 44419412 IC50 = 7289 nM T00884 CN1WA4 44419439 IC50 = 378 nM T00884 CKID29 44419441 IC50 = 1548 nM T00884 C60WDB 44419448 IC50 = 293 nM T00884 C3SAK6 44419449 IC50 = 752 nM T00884 CYBP92 44419473 IC50 = 215 nM T00884 CGT14K 44419476 IC50 = 1082 nM T00884 CU3D9L 44419477 IC50 = 187 nM T00884 C7Q2DF 44419479 IC50 = 104 nM T00884 CCS0Q9 44419480 IC50 = 192 nM T00884 CCHS37 44419482 IC50 = 100 nM T00884 CZQ7F9 44419483 IC50 = 582 nM T00884 CXYP53 44419546 IC50 = 411 nM T00884 C1T3XJ 44419555 IC50 = 22 nM T00884 CA4IH6 44419558 IC50 = 188 nM T00884 CAMQ76 44432386 IC50 = 13000 nM T00884 C3C0JF 44432391 IC50 = 13000 nM T00884 CB6J0H 44432416 IC50 = 20000 nM T00884 CY1B2H 44440858 Ki = 24 nM T00884 CN4ZL9 44440859 Ki = 123 nM T00884 CN90ZV 44440860 Ki = 379 nM T00884 C0GZB2 44440865 Ki = 7.6 nM T00884 CG01PI 44440866 Ki = 30 nM T00884 CC1Z2N 44440873 Ki = 14 nM T00884 C07WNS 44446565 IC50 = 854 nM T00884 CALE50 44446566 IC50 = 463 nM T00884 C9OW0Z 44446567 IC50 = 275 nM T00884 CGM98S 44446568 IC50 = 6062 nM T00884 CXJ51G 44446569 IC50 = 568 nM T00884 C9DCO6 44446570 IC50 = 182 nM T00884 C34XTN 44446577 IC50 = 4870 nM T00884 CW63PF 44446580 IC50 = 3376 nM T00884 C5QWB7 44446583 IC50 = 3434 nM T00884 CJZ13N 44446593 IC50 = 100 nM T00884 CEK28S 44446595 IC50 = 93 nM T00884 C7VE2J 44446596 IC50 = 150 nM T00884 C71OQP 44446598 IC50 = 526 nM T00884 CPK8T3 44446602 IC50 = 221 nM T00884 C5CAE9 44446604 IC50 = 345 nM T00884 CA0K6E 44446605 IC50 = 1023 nM T00884 C3TZV2 44446607 IC50 = 795 nM T00884 C31JGN 44446608 IC50 = 805 nM T00884 C9R2IX 44446610 IC50 = 703 nM T00884 C91YQW 44446611 IC50 = 302 nM T00884 CBLF23 44446613 IC50 = 224 nM T00884 C1N9QM 44446614 IC50 = 289 nM T00884 C54CVM 44446616 IC50 = 812 nM T00884 CB2VC0 44446617 IC50 = 165 nM T00884 C8OUJ2 44446621 IC50 = 1110 nM T00884 C6AGR1 44446631 IC50 = 1372 nM T00884 CTF63M 44446635 IC50 = 2856 nM T00884 CKGN35 44446639 IC50 = 244 nM T00884 CIDA76 44446641 IC50 = 62 nM T00884 CZ7S4Y 44446645 IC50 = 171 nM T00884 CTO73Z 44446647 IC50 = 104 nM T00884 CEZ48V 44446650 IC50 = 148 nM T00884 CON0S6 44447608 IC50 = 412 nM T00884 C8ZLV4 44564898 Ki = 100 nM T00884 C2NFZ7 44564941 Ki = 16 nM T00884 C43RSH 44564942 Ki = 5 nM T00884 CO1WZ3 44564943 Ki = 43 nM T00884 C2U9OC 44564998 Ki = 30 nM T00884 CAK9P0 44564999 Ki = 25 nM T00884 C28OAW 44565049 Ki = 22 nM T00884 C76YJU 44565051 Ki = 24 nM T00884 CP1RO6 44565052 Ki = 10 nM T00884 CG4I0V 44565098 Ki = 34 nM T00884 CHX49N 44565099 Ki = 103 nM T00884 C3LAO8 44565100 Ki = 20 nM T00884 CH8FP0 44565148 Ki = 40 nM T00884 C8HD1U 44626319 Ki = 9700 nM T00884 CQF0A4 45271150 Ki = 54 nM T00884 CTX49I 45271151 Ki = 1221 nM T00884 CIMJ26 45272042 Ki > 1000 nM T00884 CM2BA6 45272064 Ki = 2797 nM T00884 C9NR1T 45272847 Ki = 30 nM T00884 CNXJ43 45272873 Ki = 2068 nM T00884 CSP9M7 45485756 Ki > 12000 nM T00884 C3EL4C 45485757 Ki = 4100 nM T00884 C7J8IO 45485758 Ki > 12000 nM T00884 CX6ZG2 45485775 Ki = 6500 nM T00884 CKU6S2 45485784 Ki = 5200 nM T00884 CV48KD 45485788 Ki > 12000 nM T00884 CUE8N7 45485798 Ki > 12000 nM T00884 CK3N1G 46206137 IC50 > 10000 nM T00884 C0CEV2 46897163 IC50 = 31 nM T00884 C78MYC 56839292 IC50 > 5000 nM T00884 CD35UF 56839293 IC50 > 5000 nM T00884 CTFL56 56839294 IC50 = 1400 nM T00884 CYA2V8 56839499 IC50 = 681 nM T00884 CZG2O3 71720517 IC50 = 1995.26 nM T00884 C6ENV5 100951623 IC50 = 3800 nM T00884 C3YNJ7 122187254 IC50 = 611 nM T00884 CUL9I1 122187255 IC50 = 4100 nM T00884 CCD97V 122187256 IC50 = 4300 nM T00884 C6MW4Q 122187257 IC50 = 1700 nM T00884 CUFD82 122187258 IC50 > 5000 nM T00884 CHNY79 122187259 IC50 = 1340 nM T00884 C6HB2K 122187260 IC50 = 2500 nM T00884 CQ16CH 122187261 IC50 = 1700 nM T00884 CD7Z4N 122187262 IC50 = 1700 nM T00884 C9V7XK 122187263 IC50 = 326 nM T00884 CE8S4F 122187264 IC50 > 5000 nM T00884 CO5UZ9 122187265 IC50 > 5000 nM T00884 CEZ14H 122187266 IC50 = 3.3 nM T00884 CRBQ58 122187267 IC50 > 5000 nM T00884 C0VD5A 122187268 IC50 = 7 nM T00884 CQB0L1 122187269 IC50 = 2050 nM T00884 CY1S7I 122187270 IC50 > 5000 nM T00884 CF89ON 122187271 IC50 = 444 nM T00884 CBJ90L 135405057 Ki = 46 nM T00884 CW51VO 135485575 Ki = 8990 nM T00884 CL9BV0 135497124 Ki = 14 nM T00884 C7S2TQ 135539041 Ki = 5950 nM T00884 C9XUH4 135539055 Ki = 61 nM T00884 C2RDY4 135814570 Ki = 21 nM T00884 C8X7UT 135937901 Ki = 52 nM T00884 CID30V 136036234 Ki = 126 nM T00884 CI4PS1 136036235 Ki = 78 nM T00884 C7FX0N 136036236 Ki = 13 nM T00884 C1NF6Y 136036238 Ki = 35 nM T00884 CH78DC 136036240 Ki = 53 nM T00884 C0YVI5 136036241 Ki = 15 nM T00884 CME5L2 136036242 Ki = 15 nM T00884 CQ2VE9 136036243 Ki = 76 nM T00884 C5AR1O 136036244 Ki = 14 nM T00884 CRN73I 136036245 Ki = 18 nM T00884 CSL40I 136036246 Ki = 7.5 nM T00884 C3ZUN6 136036249 Ki = 38 nM T00884 COB78Q 136036250 Ki = 13 nM T00884 C2CO6U 136036251 Ki = 34 nM T00884 CNV4H2 136036252 Ki = 14 nM T00884 CA8JF5 136036253 Ki = 43 nM T00884 CR8LO7 136036254 Ki = 36 nM T00884 C6O0PW 136036255 Ki = 20 nM T00884 CI2L5T 136036256 Ki = 16 nM T00884 C6FS8C 136036257 Ki = 44 nM T00884 CXZ4F3 136036517 Ki = 2000 nM T00884 CLF7E4 136036518 Ki = 2800 nM T00884 C4FRC5 136036519 Ki = 652 nM T00884 C67PHR 136036520 Ki = 1100 nM T00884 CSK0N6 136036521 Ki = 188 nM T00884 CU4YJ8 136036522 Ki = 129 nM T00884 CAF2H5 155531736 IC50 = 2900 nM T00884 D05AZU 11184341 IC50 = 21000 nM T00884 D06WVV 11414633 IC50 = 33200 nM T00884 D09MAZ 46897162 IC50 = 903 nM T00884 D0D8LQ 9949456 IC50 = 15100 nM T00884 D0J1XP 11818139 IC50 = 46200 nM T00884 D0Q8TD 44393620 IC50 = 22 nM T00884 D0U2UJ 3618472 IC50 = 18200 nM T01283 CQOA31 44446575 IC50 = 42000 nM T01283 C3GX7H 44446576 IC50 = 75000 nM T01283 C8ZD4N 44446579 IC50 = 83000 nM T01283 CGMT57 44446585 IC50 = 48000 nM T01283 C93NGT 44446586 IC50 = 64000 nM T01283 C3X6DO 44446591 IC50 = 58000 nM T01283 CD2HI5 44446592 IC50 = 42000 nM T01283 C76IJN 44446594 IC50 = 91000 nM T01283 CE0B5D 44446599 IC50 = 93000 nM T01283 COB8L1 44446600 IC50 = 114000 nM T01283 CTOJ01 44446601 IC50 = 139000 nM T01283 CM8U9N 44446603 IC50 = 54000 nM T01283 CI7A0F 44446618 IC50 = 54000 nM T01283 COG95M 44446619 IC50 = 41000 nM T01283 CAIP09 44446620 IC50 = 27000 nM T01283 CN8K1R 44446623 IC50 = 26000 nM T01283 CY90WO 44446624 IC50 = 26000 nM T01283 CEVY78 44446628 IC50 = 30000 nM T01283 CEW06I 44446636 IC50 = 26000 nM T01283 C7BA0O 44446637 IC50 = 29000 nM T01283 CLE13Y 44446640 IC50 = 20000 nM T01283 CUP0B7 44446643 IC50 = 12000 nM T01283 C64JAX 44446646 IC50 = 13000 nM T01283 C2CNI0 44446649 IC50 = 17000 nM T01283 CL1BP6 44446653 IC50 = 21000 nM T01283 CF46DN 44446655 IC50 = 25000 nM T01283 CV17CR 44446657 IC50 = 16000 nM T01283 C83OQD 44446658 IC50 = 16000 nM T01283 CT1WV9 44446660 IC50 = 32000 nM T01283 C3XHQ7 44446661 IC50 = 30000 nM T01283 C2Y3IJ 44446663 IC50 = 27000 nM T01283 CO5W4F 44446664 IC50 = 23000 nM T01283 CC61IO 44446670 IC50 = 41000 nM T01283 CJZ3Q9 44446673 IC50 = 23000 nM T01283 CFQ89H 44446674 IC50 = 16000 nM T01283 C50BKU 44446675 IC50 = 20000 nM T01283 C1F9QJ 44446682 IC50 = 25000 nM T01283 C15ASP 44446688 IC50 = 20000 nM T01283 CQ13KB 44446692 IC50 = 15000 nM T01283 CIOY10 44446693 IC50 = 22000 nM T01283 CCN28E 44446694 IC50 = 22000 nM T01283 CI9K8H 44446695 IC50 = 18000 nM T01283 CKN8T4 44446696 IC50 = 12000 nM T01283 CDZL68 44446848 IC50 = 16000 nM T01283 C9PDZ4 44446849 IC50 = 19000 nM T01283 CG9JX7 44446850 IC50 = 11000 nM T01283 CWUH82 44446851 IC50 = 22000 nM T01283 CF3K9T 44446852 IC50 = 19000 nM T01283 CH6P2X 44446853 IC50 = 18000 nM T01283 C3OLB5 44446854 IC50 = 17000 nM T01283 CL0Z6D 57390696 Ki = 5400 nM T01283 CQP0I3 57394205 Ki = 2700 nM T01283 C8C6FQ 57397840 Ki = 8700 nM T01283 C04VXI 57403661 Ki = 2600 nM T01283 CP52YQ 73348655 IC50 = 55000 nM T01283 CI4J7T 73348656 IC50 = 43000 nM T01283 C9Y6QZ 73351742 IC50 = 21000 nM T01283 CDG78J 90663633 IC50 = 12000 nM T01283 CZ9VR4 46905990 IC50 = 13000 nM T45228 CYCA13 86763277 IC50 = 700 nM T45228 C0ZR9Q 87055830 IC50 = 3800 nM T45228 CMXZ54 122180705 IC50 = 6000 nM T45228 C43MWH 122180706 IC50 > 1000 nM T14597 D01PZD 5329098 IC50 > 100000 nM T14597 D03ZBT 11626560 IC50 > 1000 nM T14597 D05UFG 10184653 IC50 = 14 nM T14597 D06IAR 60961 IC50 ~ 1600000 nM T14597 D06XXH 11511120 IC50 = 45.7 nM T14597 D07POC 176870 IC50 = 64 nM T14597 D08CDI 208908 IC50 = 9 nM T14597 D09KTS 24821094 IC50 = 9.4 nM T14597 D09XZB 123631 IC50 = 24 nM T14597 D0E6XR 3062316 IC50 = 710 nM T14597 D0OB0F 5328940 IC50 = 2600 nM T14597 D00NYJ 42642648 IC50 = 2 nM T14597 D00RMC 6918508 IC50 = 3400 nM T14597 D00YER 25127713 IC50 = 5.3 nM T14597 D01GFX 11640390 IC50 > 10000 nM T14597 D02PGP 448965 IC50 = 40000 nM T14597 D02TUL 118115473 IC50 > 50000 nM T14597 D02UFQ 11620908 IC50 = 3 nM T14597 D03LWG 53235510 IC50 > 10000 nM T14597 D07EHV 44814409 IC50 > 10000 nM T14597 D07HPJ 11476171 IC50 > 10000 nM T14597 D0BM7M 11488320 IC50 = 14 nM T14597 D0CN9Q 9874913 IC50 = 10 nM T14597 D0E3TC 44259 IC50 = 34 nM T14597 D0G5XV 135565884 IC50 = 530 nM T14597 D0LF1U 5287969 IC50 = 15800 nM T14597 D0Q9CY 9915743 IC50 = 1 nM T14597 D0S3PO 6445562 IC50 = 1229 nM T14597 D0S5RC 3025986 IC50 > 25000 nM T14597 D0U4FF 10437018 IC50 = 22 nM T14597 D0YB3W 156414 IC50 = 30 nM T14597 D0Z4RC 24756910 IC50 = 15.7 nM T14597 D03BNU 59604787 IC50 > 3500 nM T14597 D0LF0O 135441202 IC50 = 6000 nM T14597 D02YAQ 6603857 IC50 = 16 nM T14597 D0GZ7B 5328779 IC50 = 13489.63 nM T14597 D0L5YF 5329032 IC50 > 100000 nM T14597 D0Q7HO 4705 IC50 = 5400 nM T14597 D0T3ME 156422 IC50 > 20000 nM T14597 CWC0F6 76146 IC50 = 29000 nM T14597 C63WLY 89644 IC50 > 10 ug.mL-1 T14597 C5JE2Z 104860 IC50 > 10 ug.mL-1 T14597 CRFU83 156413 IC50 = 9 nM T14597 CI1NA5 159926 IC50 = 7.3 ug.mL-1 T14597 C2P8XO 176871 IC50 = 1520 nM T14597 CYBA43 177458 IC50 > 10 ug.mL-1 T14597 CVXN37 313371 IC50 = 11400 nM T14597 CQ32PZ 331313 IC50 = 10800 nM T14597 CK0L4O 442514 IC50 = 960 nM T14597 CRYI40 448969 IC50 = 12000 nM T14597 C9D7UY 727518 IC50 > 100000 nM T14597 C6S9MF 800888 IC50 = 31000 nM T14597 CXB5A2 964113 IC50 > 100000 nM T14597 CDB17F 1538822 IC50 = 16900 nM T14597 C1P4FC 1838043 IC50 = 4897.79 nM T14597 CZ2B4M 2358462 IC50 > 100000 nM T14597 CXA1L7 2365265 IC50 > 100000 nM T14597 CEF62M 2379240 IC50 > 100000 nM T14597 CS6RH2 2385464 IC50 = 16982.44 nM T14597 CKT64G 2396126 IC50 > 10000 nM T14597 CKE7P2 2725645 IC50 = 1910 nM T14597 CG43CZ 2802451 IC50 = 3830 nM T14597 COZN45 3417197 IC50 = 18000 nM T14597 CJVK95 5076757 IC50 > 50000 nM T14597 CTID76 5282335 IC50 > 25000 nM T14597 CY28LS 5293755 IC50 > 100000 nM T14597 CQ3SK4 5328203 IC50 = 170 nM T14597 CDV19S 5328354 IC50 = 379000 nM T14597 C1D0YT 5328357 IC50 = 1100000 nM T14597 CC4O6Y 5328360 IC50 = 219000 nM T14597 CND59O 5328761 IC50 = 12882.5 nM T14597 C68MGU 5328762 IC50 = 10000 nM T14597 CN8L0R 5328764 IC50 = 12000 nM T14597 C2B0HF 5328765 IC50 = 3000 nM T14597 C4HNQ7 5328766 IC50 = 34673.69 nM T14597 CLQ73F 5328767 IC50 = 50000 nM T14597 C3F7YW 5328770 IC50 = 34673.69 nM T14597 C67KXB 5328771 IC50 = 42000 nM T14597 CJ6U2C 5328773 IC50 = 22908.68 nM T14597 C7VW9X 5328774 IC50 = 57000 nM T14597 CSL05I 5328775 IC50 > 500000 nM T14597 C5ZV9K 5328776 IC50 = 331131.12 nM T14597 CI97TH 5328778 IC50 = 165958.69 nM T14597 CMX61C 5328780 IC50 = 49000 nM T14597 CED31Y 5328781 IC50 = 33884.42 nM T14597 CT1QC6 5328954 IC50 = 14 nM T14597 C41BJK 5328955 IC50 = 38 nM T14597 CUW4V3 5328956 IC50 = 177 nM T14597 CI3Q6X 5328957 IC50 = 113 nM T14597 C0AF9T 5328958 IC50 = 162 nM T14597 C8A4XJ 5328959 IC50 = 85 nM T14597 CTN9X5 5328960 IC50 = 73 nM T14597 CP6G8R 5328961 IC50 = 53 nM T14597 CAQM41 5328962 IC50 = 124 nM T14597 CDJ8B5 5328964 IC50 = 183 nM T14597 C94KSU 5328965 IC50 = 33 nM T14597 C1W0DS 5328966 IC50 = 116 nM T14597 CX5S2M 5328967 IC50 = 9 nM T14597 CHL05B 5328968 IC50 = 16 nM T14597 CXN2Y0 5328969 IC50 = 301 nM T14597 C6BM9P 5328970 IC50 = 1164 nM T14597 CR3GV8 5328971 IC50 = 1428 nM T14597 CJU57A 5328972 IC50 = 1559 nM T14597 CJ42FQ 5328973 IC50 = 2776 nM T14597 CKA09Y 5328974 IC50 = 2808 nM T14597 C92KTO 5328975 IC50 = 1912 nM T14597 C4KI5U 5328976 IC50 = 733 nM T14597 CI36GZ 5328977 IC50 = 634 nM T14597 CU4W7S 5328978 IC50 = 414 nM T14597 C39VSH 5328979 IC50 = 1592 nM T14597 C9U5YF 5328980 IC50 = 15624 nM T14597 CY4B5J 5328981 IC50 = 15238 nM T14597 C03WIS 5328982 IC50 = 91325 nM T14597 CG3KL4 5328983 IC50 = 8832 nM T14597 CV5KY4 5328984 IC50 = 5042 nM T14597 CUJ6G5 5328985 IC50 = 458 nM T14597 CLP07T 5328986 IC50 = 25710 nM T14597 CD60RC 5328987 IC50 = 4182 nM T14597 CK15AU 5328988 IC50 = 21657 nM T14597 C7R2EK 5328989 IC50 = 2921 nM T14597 CFW19M 5329009 IC50 = 24 nM T14597 CH26SN 5329069 IC50 = 3.9 nM T14597 C5JL2Y 5329085 IC50 = 110 nM T14597 CT4U5F 5329086 IC50 = 207 nM T14597 CBY4R5 5329087 IC50 = 13 nM T14597 C53HOJ 5329088 IC50 = 14 nM T14597 C2P3EO 5329089 IC50 = 5 nM T14597 C61NGH 5329090 IC50 = 8.1 nM T14597 CAV71E 5329092 IC50 = 24 nM T14597 CTQ18A 5329232 IC50 = 300 nM T14597 CQG6R2 5329234 IC50 > 5000 nM T14597 CPS7X1 5329236 IC50 = 100 nM T14597 C41UBI 5329239 IC50 = 400 nM T14597 C6VQ9F 5329240 IC50 = 200 nM T14597 C6PJ2R 5329243 IC50 = 100 nM T14597 C0OKB7 5329244 IC50 = 200 nM T14597 C78ZNL 5329245 IC50 = 500 nM T14597 CK8FH6 5329249 IC50 = 2780 nM T14597 CN5B6C 5329250 IC50 = 100 nM T14597 CQ0B6E 5329251 IC50 = 100 nM T14597 C4KO3N 5329252 IC50 = 40 nM T14597 CQ39FM 5329480 IC50 = 10 nM T14597 CVS3Z1 5329481 IC50 = 263 nM T14597 CW2UJ7 5329482 IC50 = 977 nM T14597 CY14AK 5329483 IC50 = 95 nM T14597 CIT24W 5329484 IC50 = 309 nM T14597 CDZ6R5 5329485 IC50 = 347 nM T14597 C3LSH8 5329486 IC50 = 234 nM T14597 CGZA12 5329487 IC50 = 1778 nM T14597 CV9L1J 5329488 IC50 = 117 nM T14597 CJD92I 5329489 IC50 = 234 nM T14597 CS1HF6 5329490 IC50 = 210 nM T14597 CX4L0Q 5329491 IC50 = 147 nM T14597 C9C3SD 5329492 IC50 = 10 nM T14597 CDRM58 5329493 IC50 = 19 nM T14597 CUCE63 5329663 IC50 > 25000 nM T14597 CB0QZ2 5330117 IC50 > 1000 nM T14597 C7QZL3 5330118 IC50 > 1000 nM T14597 CNR9B8 5330119 IC50 > 1000 nM T14597 CXY2I9 5330120 IC50 > 1000 nM T14597 CDF96J 5330121 IC50 > 1000 nM T14597 C7BPR2 5330122 IC50 > 1000 nM T14597 CC4ZJ3 5330123 IC50 > 1000 nM T14597 CLV0T6 5330124 IC50 > 1000 nM T14597 CUEZ35 5330437 IC50 = 2500 nM T14597 C3U0TG 5330830 IC50 > 100000 nM T14597 CL1FH5 5330832 IC50 > 100000 nM T14597 C1P2ZA 5330847 IC50 > 100000 nM T14597 CYXI29 5353388 IC50 = 37153.52 nM T14597 CDQ3M7 5359485 IC50 = 9.4 ug.mL-1 T14597 C54BYP 5360741 IC50 = 4.5 ug.mL-1 T14597 CD65JT 5427216 IC50 > 100000 nM T14597 CPB95V 5427224 IC50 = 22500 nM T14597 CA6L5V 5707304 IC50 > 100000 nM T14597 C43YGE 5713379 IC50 > 100000 nM T14597 CT8U7I 5874584 IC50 > 100000 nM T14597 CM8LW9 6036100 IC50 > 100000 nM T14597 C7MD9J 6091659 IC50 = 346.74 nM T14597 CO5SZ1 6440837 IC50 > 200 ug.mL-1 T14597 CTB7N5 6447926 IC50 = 128.82 nM T14597 CQ3S8L 6450842 IC50 > 100000 nM T14597 CW5YJ2 6536705 IC50 > 100000 nM T14597 C2B4ZE 9803006 IC50 = 2120 nM T14597 CF47BP 9806229 IC50 = 19 nM T14597 C72WMK 9808725 IC50 = 360 nM T14597 CZ2MH9 9809611 IC50 = 30 nM T14597 CNJE78 9811391 IC50 = 100 nM T14597 CZ5VX6 9820644 IC50 = 73 nM T14597 CRKD07 9825976 IC50 = 27 nM T14597 C4XU5Z 9828336 IC50 = 26 nM T14597 C5S8FR 9829680 IC50 = 18 nM T14597 CYWI50 9830092 IC50 = 200 nM T14597 CBGE59 9833337 IC50 = 7000 nM T14597 CGKC15 9851149 IC50 = 90 nM T14597 C41QWA 9857146 IC50 > 10000 nM T14597 CN1F9T 9858558 IC50 = 21000 nM T14597 CM5Z8X 9869943 IC50 > 10000 nM T14597 C12PKF 9871380 IC50 = 40 nM T14597 C2FW1X 9872621 IC50 = 22 nM T14597 CS51KJ 9873631 IC50 = 100 nM T14597 CU2N8D 9873657 IC50 = 24 nM T14597 C5NK9U 9873849 IC50 = 22 nM T14597 C5CLD8 9874613 IC50 = 141 nM T14597 CUZ07T 9884745 IC50 = 64800 nM T14597 C2JR8Q 9887521 IC50 = 3870 nM T14597 CXL31W 9890154 IC50 = 4490 nM T14597 CIN0E2 9891993 IC50 = 31430 nM T14597 CXA5C8 9893493 IC50 = 5300 nM T14597 CE87TX 9893671 IC50 = 31 nM T14597 CEJ05V 9894581 IC50 = 17 nM T14597 C4WQK8 9897300 IC50 = 6.4 nM T14597 CB4DT1 9899125 IC50 = 58884.37 nM T14597 CMKX01 9906303 IC50 = 16000 nM T14597 C01WSX 9907221 IC50 = 1.9 nM T14597 C9SQU4 9913648 IC50 = 2970 nM T14597 CF3KI0 9917474 IC50 = 28 nM T14597 C67BSM 9919900 IC50 = 60 nM T14597 CYW49X 9927718 IC50 > 25000 nM T14597 CWT56C 9930439 IC50 = 1630 nM T14597 CP2J4W 9930632 IC50 = 7.6 nM T14597 CO85KA 9932061 IC50 = 250 nM T14597 CPYB98 9934935 IC50 = 7800 nM T14597 CU56DE 9937225 IC50 = 21 nM T14597 CLT0U5 9937660 IC50 = 23 nM T14597 CS5KX9 9938299 IC50 > 10000 nM T14597 CXJR73 9938805 IC50 = 141 nM T14597 C6HP3L 9948410 IC50 = 92600 nM T14597 C06JHE 9952784 IC50 = 50 nM T14597 CI51BV 9954075 IC50 = 1950 nM T14597 CBE9O6 9954156 IC50 = 30 nM T14597 C0ZO2V 9960493 IC50 = 26 nM T14597 CSU19Y 9960734 IC50 = 20 nM T14597 CHD79R 9969008 IC50 = 4.2 nM T14597 C24MZU 9974694 IC50 = 4.3 nM T14597 CROV41 9979362 IC50 = 11750 nM T14597 CH03DY 9984664 IC50 = 33950 nM T14597 CO4N3Q 9995374 IC50 = 13200 nM T14597 CQX39R 10006530 IC50 = 1692 nM T14597 CO2PA9 10029703 IC50 = 23590 nM T14597 C7YD1X 10048045 IC50 > 25000 nM T14597 CK8RL4 10071409 IC50 = 30 ug.mL-1 T14597 C1JUF8 10073832 IC50 > 10000 nM T14597 CC0J9E 10075664 IC50 = 26 nM T14597 C35HXN 10085225 IC50 = 45000 nM T14597 CF09NK 10098235 IC50 = 34130 nM T14597 CZ9Y1G 10106867 IC50 = 2070 nM T14597 C5SV9C 10114464 IC50 = 60 nM T14597 C80ZDK 10115240 IC50 = 81 nM T14597 C7C1IG 10116123 IC50 = 76 nM T14597 CMK79O 10117051 IC50 = 76 nM T14597 C0RV4A 10140801 IC50 = 360 nM T14597 CREM37 10151881 IC50 = 22 nM T14597 CC4X6M 10152238 IC50 < 2 nM T14597 C5HB2P 10152514 IC50 = 31 nM T14597 C14ZEP 10156890 IC50 = 12180 nM T14597 CUD7L1 10159833 IC50 = 47 nM T14597 CA40TZ 10161969 IC50 = 380 nM T14597 CHU9C6 10162630 IC50 < 2 nM T14597 CK4OH0 10162954 IC50 < 2 nM T14597 CGW26V 10163178 IC50 = 14 nM T14597 CU9SK6 10183346 IC50 = 280 nM T14597 CQP8Y1 10194801 IC50 = 90 nM T14597 CI4Q0J 10195479 IC50 = 70 nM T14597 C47FXG 10200918 IC50 = 6880 nM T14597 C5YCN2 10215023 IC50 > 100000 nM T14597 CNTU23 10217083 IC50 = 70 nM T14597 CSGL59 10217304 IC50 = 120 nM T14597 CEW30I 10217590 IC50 = 55 nM T14597 C67POS 10223065 IC50 = 4500 nM T14597 CCVU79 10226418 IC50 = 130 nM T14597 C2KSD3 10227095 IC50 = 200 nM T14597 C6QP4E 10227907 IC50 = 54 nM T14597 CPD6Z9 10236164 IC50 > 100000 nM T14597 C1UB5A 10253204 IC50 = 4160 nM T14597 CBI47E 10264222 IC50 > 100000 nM T14597 CE68KY 10277546 IC50 = 370 nM T14597 C9K0SA 10288761 IC50 < 2 nM T14597 CJ4D9B 10288917 IC50 = 750 nM T14597 CNU74Z 10288918 IC50 = 39 nM T14597 CCE64Z 10288920 IC50 = 38 nM T14597 C8NMA6 10295839 IC50 = 4680 nM T14597 C7SFI1 10296883 IC50 > 10000 nM T14597 CVO54Z 10300451 IC50 = 40 nM T14597 CGF21D 10310843 IC50 = 63 nM T14597 CEN48D 10322889 IC50 = 5660 nM T14597 CVP85S 10385997 IC50 > 500 nM T14597 CEXH09 10405907 IC50 = 4400 nM T14597 C32REN 10411907 IC50 = 46 nM T14597 CQ43JU 10426229 IC50 = 7000 nM T14597 C2SXE3 10430383 IC50 = 251.19 nM T14597 CC5OM4 10473589 IC50 > 200 ug.mL-1 T14597 C7PLI5 10478569 IC50 = 8000 nM T14597 CU3A8H 10484995 Ki = 30000 nM T14597 CJWH60 10489322 IC50 > 100000 nM T14597 C09NYR 10507839 IC50 = 5.9 ug.mL-1 T14597 CLH12I 10523411 IC50 = 125 nM T14597 C38RSF 10528818 IC50 = 12 nM T14597 C5SVT4 10537949 IC50 > 100000 nM T14597 C7JX3G 10547930 IC50 = 8.6 nM T14597 CGAW17 10562306 IC50 > 100000 nM T14597 C6AJI9 10562777 IC50 > 100000 nM T14597 CE5L6D 10587839 IC50 > 100000 nM T14597 CM8N6L 10593765 IC50 > 100000 nM T14597 CI30LZ 10613858 IC50 > 100000 nM T14597 CTG7H5 10614224 IC50 = 10780 nM T14597 CT0O5K 10634145 IC50 > 50 ug.mL-1 T14597 CH6Z3L 10635478 IC50 > 100000 nM T14597 CB97UD 10636005 IC50 > 100000 nM T14597 C2UWA0 10658651 IC50 > 100000 nM T14597 C64DFG 10662351 IC50 = 8.8 nM T14597 C5L0IX 10663368 IC50 > 100000 nM T14597 C9Z7XH 10663503 IC50 = 66600 nM T14597 CFGL61 10672994 IC50 = 182 nM T14597 CDV84T 10673774 IC50 = 8.2 nM T14597 CH1G6P 10682457 IC50 > 100000 nM T14597 C51VNS 10691590 IC50 = 7.3 nM T14597 C6BK7Q 10691652 IC50 = 1.1 nM T14597 C54UAK 10728035 IC50 > 100000 nM T14597 CN8GS6 10738988 IC50 = 26 nM T14597 CXSH91 10753550 IC50 > 100000 nM T14597 CVPW04 10755069 IC50 > 100000 nM T14597 CYAL86 10759828 IC50 = 3 nM T14597 C3WR0Q 10779668 IC50 = 91400 nM T14597 CF5T1H 10783444 IC50 = 16200 nM T14597 C62FWK 10791534 IC50 > 200 nM T14597 CK2ZP3 10805953 IC50 > 50 ug.mL-1 T14597 CX2E1C 10829071 IC50 = 670 nM T14597 CWX4V1 10838598 IC50 > 5000 nM T14597 C01KXI 10854884 IC50 = 12 nM T14597 CTI84S 10884588 IC50 = 300 nM T14597 C7DK8H 10885120 IC50 = 4390 nM T14597 CP5XT0 10906920 IC50 = 180 nM T14597 CBM57K 10918242 IC50 = 33950 nM T14597 CIRP84 10928765 IC50 = 11820 nM T14597 CI01XA 10951285 IC50 = 4130 nM T14597 CEKW21 10972694 IC50 = 1210 nM T14597 C1I6VX 10973080 IC50 = 9580 nM T14597 CTY19K 10973186 IC50 = 320 nM T14597 COE13S 10983483 IC50 = 8740 nM T14597 C2AK4W 11005320 IC50 = 450 nM T14597 CM4JD2 11037303 IC50 = 21510 nM T14597 CR91TM 11102890 IC50 = 9350 nM T14597 C8TA4Z 11129889 IC50 > 100000 nM T14597 COB20T 11157041 IC50 = 1134 nM T14597 CUIX38 11157794 IC50 = 28 nM T14597 C0VD5M 11168387 IC50 = 498 nM T14597 CSZ6B2 11168731 IC50 = 8100 nM T14597 CQ7PU5 11178756 IC50 = 22 nM T14597 C7XU5W 11180271 IC50 = 39 nM T14597 C9Z6AG 11180494 IC50 = 625 nM T14597 CHV1P9 11180599 IC50 = 2100 nM T14597 C2B7HJ 11180905 IC50 = 25 nM T14597 CRG7B6 11192261 IC50 = 131 nM T14597 CA6L9Y 11192678 IC50 = 59 nM T14597 C2PMR9 11192753 IC50 = 18 nM T14597 CA07YO 11193143 IC50 = 3775 nM T14597 C0K8NB 11202869 IC50 = 800 nM T14597 C6N8EO 11203411 IC50 = 20 nM T14597 C16HXD 11203436 IC50 = 61 nM T14597 C7H8AD 11203663 IC50 = 83 nM T14597 C87QSN 11203886 IC50 = 76 nM T14597 C1YB7C 11220978 IC50 = 9 nM T14597 CNZ2H8 11226874 IC50 = 26000 nM T14597 CMZ8S5 11227115 IC50 = 10 nM T14597 C2W5RC 11235063 IC50 > 50000 nM T14597 C98HRX 11237508 IC50 = 363 nM T14597 CXN98V 11238293 IC50 = 269 nM T14597 CSX6P5 11238512 IC50 = 33 nM T14597 CWOU43 11238694 IC50 = 81 nM T14597 CG07FL 11238864 IC50 = 540 nM T14597 C0QN4V 11238875 IC50 = 196 nM T14597 CU27LB 11246488 IC50 = 143 nM T14597 CGP6U2 11249521 IC50 = 3781 nM T14597 CO97YK 11249776 IC50 = 62 nM T14597 CJ02WR 11249881 IC50 = 246 nM T14597 CWG8Y6 11271094 IC50 = 208 nM T14597 C5ZKN4 11271821 IC50 = 89 nM T14597 CIW3X5 11272368 IC50 = 46 nM T14597 CR35NY 11273032 IC50 = 10 nM T14597 C6C3JX 11281930 IC50 > 10000 nM T14597 CUO27S 11282791 IC50 > 500 nM T14597 C5EO4X 11284905 IC50 = 83 nM T14597 CJ6R3N 11284937 IC50 = 50 nM T14597 CIV3Y6 11285080 IC50 = 58 nM T14597 CSN45Y 11289919 IC50 = 120000 nM T14597 CBOP58 11293798 Ki > 10000 nM T14597 CH02JX 11296170 IC50 = 161 nM T14597 C5Z6NC 11296256 IC50 = 406 nM T14597 CU9ER4 11296411 IC50 = 1184 nM T14597 C80IVP 11305772 IC50 = 96 nM T14597 CLP14E 11306338 IC50 = 120 nM T14597 CP3BM8 11307161 IC50 = 2600 nM T14597 C18BHK 11307255 IC50 = 184 nM T14597 C64SCF 11307581 IC50 = 10 nM T14597 C6OQC2 11307602 IC50 = 40 nM T14597 CZN3Q6 11307866 IC50 = 25 nM T14597 CK91YW 11317404 IC50 = 100 nM T14597 CN2P4G 11328571 IC50 = 60 nM T14597 CT7CG8 11341400 IC50 = 13200 nM T14597 CXI48D 11342107 IC50 = 281 nM T14597 C8FQY5 11342284 IC50 = 44 nM T14597 CO2E6V 11342331 IC50 = 8 nM T14597 CLA1W0 11342405 IC50 = 89 nM T14597 C3KC4P 11353443 IC50 = 76 nM T14597 C49AZU 11354013 IC50 = 29 nM T14597 CDZR14 11357877 IC50 > 1000 nM T14597 C26BZX 11362471 Ki > 10000 nM T14597 C7QNX8 11363138 IC50 = 162 nM T14597 CK14GM 11365122 IC50 = 132 nM T14597 C3BMQ0 11365185 IC50 = 7 nM T14597 C5WI2V 11365297 IC50 = 27 nM T14597 CX5FE9 11365342 IC50 = 24 nM T14597 CYF58P 11365726 IC50 = 13 nM T14597 C8OW4X 11375205 IC50 = 220 nM T14597 CN4O0Q 11376079 IC50 = 1477 nM T14597 CT3W2J 11376208 IC50 = 15 nM T14597 C10XFS 11382411 IC50 = 7 nM T14597 C3WYU1 11387244 IC50 = 230 nM T14597 CWXB93 11397177 Ki > 10000 nM T14597 C8F0BE 11397750 IC50 = 100 nM T14597 CW42QJ 11398239 IC50 = 91 nM T14597 CA9N1G 11398437 IC50 = 1055 nM T14597 CN4WA3 11398461 IC50 = 75 nM T14597 CBV84Q 11398999 IC50 = 78 nM T14597 C2V7RQ 11399289 IC50 = 20 nM T14597 CY76XJ 11399310 IC50 = 74 nM T14597 C6UXH4 11399331 IC50 = 64 nM T14597 CV5IR8 11410608 IC50 = 69 nM T14597 C9N3PO 11410634 IC50 = 9800 nM T14597 CG7ES9 11410940 IC50 = 169 nM T14597 C94QJA 11420204 IC50 = 13 nM T14597 C1I4JO 11421443 IC50 = 155 nM T14597 CTCG60 11421783 IC50 = 732 nM T14597 CU6FD4 11421877 IC50 = 2100 nM T14597 C0KWX9 11422340 IC50 = 104 nM T14597 C5KWS9 11422548 IC50 = 603 nM T14597 C7AI2V 11432911 IC50 > 25000 nM T14597 CYD2A6 11440253 IC50 = 6 nM T14597 C3PFX4 11444623 IC50 = 59 nM T14597 CXV39N 11444862 IC50 = 1331 nM T14597 CWI62M 11454712 IC50 = 4 nM T14597 C4LZ0F 11455794 IC50 = 28 nM T14597 CFHP63 11456360 IC50 = 1134 nM T14597 CZBF91 11476645 IC50 = 226 nM T14597 C4NR5C 11477567 IC50 = 310 nM T14597 C6M9NC 11477626 IC50 > 10000 nM T14597 CD8RQ7 11478340 IC50 = 348 nM T14597 CVFE14 11478925 IC50 = 183 nM T14597 C62KHL 11489786 IC50 = 103 nM T14597 CG7XZ1 11490270 IC50 = 50 nM T14597 CKU96Z 11490477 IC50 = 1391 nM T14597 C6-AUG 11496207 IC50 = 36 nM T14597 CQA23N 11496987 IC50 = 35 nM T14597 C40GHQ 11502866 IC50 = 780 nM T14597 CLWG73 11502887 IC50 = 140 nM T14597 CJ05GR 11503005 IC50 = 180 nM T14597 C08APU 11503073 IC50 = 300 nM T14597 C3QCI7 11504234 IC50 = 100 nM T14597 C84KRP 11512802 IC50 = 90 nM T14597 CH2IZ9 11517688 IC50 = 5000 nM T14597 CU13WV 11518389 IC50 = 0.7 nM T14597 C91JCX 11518627 IC50 = 3 nM T14597 CF0YW7 11518637 IC50 = 464 nM T14597 CJGE43 11519125 IC50 = 140 nM T14597 CV3NK7 11524106 IC50 = 5.4 nM T14597 CQ63ER 11524582 IC50 > 63 nM T14597 CI5ET2 11525434 IC50 = 38 nM T14597 CL7X4Q 11530963 IC50 = 50000 nM T14597 CT75DZ 11532242 IC50 = 2.6 nM T14597 CD8SQ6 11533311 IC50 = 120 nM T14597 C1SGF3 11533556 IC50 = 4 nM T14597 CTG83F 11539329 Ki > 1400 nM T14597 C5VO2C 11539461 IC50 = 22 nM T14597 C4SNI6 11542889 IC50 > 10000 nM T14597 CG16ZV 11547377 IC50 = 130 nM T14597 CM8JD2 11547919 IC50 = 140 nM T14597 CLBH14 11547991 IC50 = 6 nM T14597 C0X4NI 11548875 IC50 = 180 nM T14597 CX6KD1 11553647 IC50 = 46 nM T14597 CPT4K5 11554463 IC50 = 3060 nM T14597 CYA8U7 11556271 IC50 = 210 nM T14597 C3MD0B 11557040 IC50 = 5 nM T14597 CI50OC 11558284 IC50 = 890 nM T14597 CB46CA 11561058 IC50 = 60 nM T14597 CS2U5G 11561468 IC50 = 47 nM T14597 CXT51U 11561779 IC50 = 2 nM T14597 C5MK1Z 11562650 IC50 = 350 nM T14597 CQ8CJ9 11562662 IC50 = 19 nM T14597 CZ2RO8 11567291 IC50 = 8000 nM T14597 CKUR82 11568720 IC50 = 0.8 nM T14597 CNV08X 11569158 IC50 < 1 nM T14597 C2R0XV 11569434 IC50 = 17 nM T14597 CO8UB2 11569903 IC50 = 2 nM T14597 C5EJ7I 11574041 IC50 = 3500 nM T14597 CU3Q1T 11576231 IC50 = 13 nM T14597 C8JW7U 11577059 IC50 = 79 nM T14597 CP25VI 11581013 IC50 = 20000 nM T14597 CA74QZ 11581908 IC50 = 1580 nM T14597 CXMY21 11583563 IC50 = 160 nM T14597 C8ZHL0 11589515 IC50 = 5400 nM T14597 CMIL86 11590363 Ki > 1400 nM T14597 CN31OR 11590557 IC50 = 2.3 nM T14597 CCPK51 11590799 IC50 = 26 nM T14597 CK4E6V 11591222 IC50 = 2 nM T14597 CR06MA 11595844 IC50 = 2.1 nM T14597 CHZ38O 11597061 IC50 = 3 nM T14597 CP1O4N 11597180 IC50 = 55 nM T14597 CR1FG0 11604864 IC50 = 2 nM T14597 CC48BK 11605761 IC50 = 52 nM T14597 CFEK68 11606101 IC50 < 1 nM T14597 CF7P3R 11611500 IC50 = 1770 nM T14597 C7TA0C 11612021 IC50 = 44 nM T14597 C9T3VC 11613187 IC50 = 0.5 nM T14597 C0T4OV 11613386 IC50 = 210 nM T14597 CSKW87 11617204 IC50 = 1890 nM T14597 CUDZ17 11619812 IC50 = 200 nM T14597 CJ73BI 11619909 IC50 = 43 nM T14597 CO68CD 11619972 IC50 < 1 nM T14597 CJ6NA8 11620487 IC50 < 1 nM T14597 C5KHN0 11625514 IC50 = 200 nM T14597 CGX96V 11626927 IC50 < 10000 nM T14597 C1VOW6 11627264 IC50 = 59 nM T14597 CQK9C3 11627337 IC50 < 1 nM T14597 CG0K4A 11632391 IC50 = 3.8 nM T14597 CK34LS 11632737 IC50 > 50000 nM T14597 CB4YR6 11634425 IC50 = 320 nM T14597 C19LFT 11634645 IC50 = 1 nM T14597 CW5A2S 11640889 IC50 = 12 nM T14597 C9T6SC 11640926 Ki > 1400 nM T14597 CA8X1L 11655791 IC50 = 69 nM T14597 C1AX2K 11656050 IC50 = 13 nM T14597 C79EDK 11657332 IC50 = 9 nM T14597 C59AXH 11663284 IC50 < 1 nM T14597 C1ZAE8 11669455 IC50 = 36 nM T14597 C5QM4L 11670167 IC50 = 5 nM T14597 C9YK5E 11675213 IC50 = 1350 nM T14597 CDA46H 11675978 IC50 = 4 nM T14597 C0MJ1S 11676469 IC50 = 5000 nM T14597 CAWX10 11677510 IC50 = 78 nM T14597 C75CNZ 11678194 IC50 = 2.9 nM T14597 C0YOG3 11681189 IC50 > 10000 nM T14597 CQ69CR 11683171 IC50 = 680 nM T14597 C9YA5W 11683816 IC50 = 1150 nM T14597 C7H9ZT 11684096 IC50 = 2 nM T14597 CQA9W7 11684098 IC50 = 36 nM T14597 CS6GJ2 11684629 IC50 = 5.1 nM T14597 C1P8JC 11684684 IC50 < 1 nM T14597 C6QI9A 11698674 IC50 = 32 nM T14597 CKF8X5 11698913 IC50 = 5 nM T14597 C5J8NA 11703562 IC50 = 231 nM T14597 CH5B6O 11705343 IC50 = 66 nM T14597 CI7O1T 11706282 IC50 < 2 nM T14597 CXOF82 11711590 IC50 = 116 nM T14597 CLY3T0 11712237 IC50 < 1 nM T14597 CWX07A 11712609 IC50 = 11 nM T14597 C93EKF 11712721 IC50 = 18 nM T14597 C4YWU2 11713043 IC50 = 0.5 nM T14597 CR51YI 11717370 IC50 = 2100 nM T14597 C8WQ9F 11719423 IC50 = 2.8 nM T14597 CC3XP1 11720499 IC50 = 69 nM T14597 CQ3R5E 11733863 IC50 = 370 nM T14597 C4HD9K 11751106 IC50 = 99 nM T14597 CKSG91 11751343 IC50 = 1700 nM T14597 CFT81W 11751635 IC50 = 1 nM T14597 C89XLW 11752667 IC50 = 18 nM T14597 C43NTX 11762902 IC50 = 1040 nM T14597 C14YAN 11786150 IC50 = 19 nM T14597 CV2RD0 11786660 IC50 = 388 nM T14597 CTZ60E 11786930 IC50 = 1000 nM T14597 CJPT37 11799155 IC50 = 189 nM T14597 C0A4TX 11955109 IC50 = 18 nM T14597 CESM43 11955112 IC50 = 36 nM T14597 CAGY67 11955434 IC50 = 74 nM T14597 C7PGH6 12175099 IC50 = 53500 nM T14597 C5MI4N 14246200 IC50 = 1130 nM T14597 CXPU45 14246203 IC50 = 1460 nM T14597 C05MWB 14738184 IC50 = 40000 nM T14597 CDGF78 15282555 IC50 = 2100 nM T14597 C7LB4I 15949613 IC50 > 10000 nM T14597 CFPW41 16007116 Ki > 1400 nM T14597 C8W6MP 16036788 IC50 = 51 nM T14597 CD51GI 16108939 IC50 = 18 nM T14597 C5YVB0 16108940 IC50 = 140 nM T14597 CBW71J 16108942 IC50 = 300 nM T14597 CG6R9L 16108943 IC50 = 92 nM T14597 CN62KM 16108944 IC50 = 230 nM T14597 C7YS5Q 16108947 IC50 = 52 nM T14597 CLD2Y4 16108948 IC50 = 1000 nM T14597 CJR95O 16108949 IC50 = 160 nM T14597 CRQ26L 16108950 IC50 = 280 nM T14597 CH80AG 16108951 IC50 = 13 nM T14597 CWB0G9 16108952 IC50 = 160 nM T14597 CZC0H1 16116961 IC50 = 8 nM T14597 CK3RG2 16116962 IC50 = 80 nM T14597 CWMO89 16116963 IC50 = 59 nM T14597 C6E8ML 16117085 IC50 = 32 nM T14597 C2ZL9X 16117347 IC50 = 230 nM T14597 C5S1YO 16117348 IC50 = 8 nM T14597 CK9T8U 16117349 IC50 = 26 nM T14597 CH3A8J 16117483 IC50 = 6 nM T14597 CO15PA 16117623 IC50 = 24 nM T14597 C4W8QZ 16117758 IC50 = 140 nM T14597 CA7I0X 16117890 IC50 = 160 nM T14597 CWA1D5 16117891 IC50 = 130 nM T14597 CBUX19 16118034 IC50 = 140 nM T14597 C1IP7J 16118035 IC50 = 57 nM T14597 C8P3XV 16118179 IC50 = 22 nM T14597 CS2AT3 16118309 IC50 = 240 nM T14597 C6D8MB 16118310 Ki = 2.7 nM T14597 C7CW9B 16118312 IC50 = 12 nM T14597 CL5IF2 16214946 IC50 > 30000 nM T14597 CU56EW 16664858 IC50 > 10000 nM T14597 CHZ20P 16730263 IC50 = 40 nM T14597 CIPX14 16736274 IC50 = 11 nM T14597 CN8WX3 16757526 IC50 = 2000 nM T14597 CQY57T 17747104 IC50 = 204 nM T14597 C4BQ6L 17747105 IC50 = 12 nM T14597 CKU29X 17747134 IC50 = 18 nM T14597 C5YZ9V 17747138 IC50 = 153 nM T14597 C95LWR 17747139 IC50 = 7 nM T14597 CW61OK 17747208 IC50 = 173 nM T14597 CQ7RH3 17747242 IC50 = 27 nM T14597 CXD23O 17747243 IC50 = 557 nM T14597 C2VL8S 17747279 IC50 = 435 nM T14597 C8AM0W 17747280 IC50 = 95 nM T14597 CEG7O8 17747281 IC50 = 25 nM T14597 CR4PF2 17747282 IC50 = 22 nM T14597 CYB3N5 17747309 IC50 = 44 nM T14597 CC2W0F 17747311 IC50 = 30 nM T14597 CS9O2H 17747339 IC50 = 76 nM T14597 CL83TA 17747341 IC50 = 189 nM T14597 C1VC9E 17747343 IC50 = 6 nM T14597 C7Q0ZD 17747376 IC50 = 255 nM T14597 CNRV46 17747535 IC50 = 470 nM T14597 CM2HS9 18176200 IC50 = 2.4 nM T14597 C7R5VZ 18967573 IC50 = 56 nM T14597 C5EH9K 20817080 IC50 = 4030 nM T14597 C3AI0N 20817111 IC50 = 200 nM T14597 C17GAL 20819668 IC50 = 264 nM T14597 C81ALS 21080010 IC50 = 50 nM T14597 CH4B5K 21081523 IC50 > 5000 nM T14597 CEBF05 21697320 IC50 = 1220 nM T14597 C82YMB 21774110 IC50 = 8 ug.mL-1 T14597 C5B7WP 21874200 IC50 = 4 nM T14597 CBN19I 21874228 IC50 = 34 nM T14597 CLD73T 21874248 IC50 = 6 nM T14597 CYSR48 21874287 IC50 = 5 nM T14597 CWY6T7 21874402 IC50 = 20 nM T14597 C5IBJ0 21874410 IC50 = 4 nM T14597 CM3XF9 21874431 IC50 = 6 nM T14597 CRB1V5 21945809 IC50 = 730 nM T14597 CT9LP3 21945841 IC50 = 500 nM T14597 C5GIE9 21945968 IC50 = 5800 nM T14597 CHU2Z3 21951965 IC50 = 220 nM T14597 CLN2G9 21952043 IC50 = 25 nM T14597 CIM14K 21952114 IC50 = 1 nM T14597 CREC34 22011954 IC50 = 4 nM T14597 CQEN87 22055240 IC50 = 60 nM T14597 C8J9GH 22055262 IC50 = 41 nM T14597 C2RY4D 22055269 IC50 = 430 nM T14597 CH5V2Q 22390479 IC50 = 120 nM T14597 C1IU0K 22390480 IC50 = 610 nM T14597 C50SLD 22390490 IC50 = 560 nM T14597 C7GK1A 22390495 IC50 = 120 nM T14597 CKV0J5 22390502 IC50 = 360 nM T14597 C5NVM0 22390522 IC50 = 110 nM T14597 C9G5RQ 22390524 IC50 = 43 nM T14597 CHF3A0 22390530 IC50 = 110 nM T14597 CD5GI0 22390536 IC50 = 110 nM T14597 C18CUK 22390541 IC50 = 190 nM T14597 C3H4NO 22390542 IC50 = 110 nM T14597 CNMZ85 22390556 IC50 = 180 nM T14597 CWL0O9 22466767 IC50 = 14700 nM T14597 C9QLP0 23133323 IC50 > 20000 nM T14597 CJ93WL 23149451 IC50 = 200 nM T14597 C39INL 23427375 IC50 = 4 ug.mL-1 T14597 CV8P7G 23546054 IC50 > 40000 nM T14597 C9PF3L 23546055 IC50 = 590 nM T14597 C2XRV0 23546056 IC50 = 1000 nM T14597 CWU9P6 23589545 IC50 = 180 nM T14597 CEN3B8 23589555 IC50 = 1200 nM T14597 C19TLD 23644675 IC50 = 680 nM T14597 CX32IF 23646535 IC50 = 2800 nM T14597 C4Z5YE 23646536 IC50 = 3000 nM T14597 CZ6E5P 23646537 IC50 = 3300 nM T14597 CG7F1M 23646539 IC50 = 820 nM T14597 C9ZSO0 23646540 IC50 = 390 nM T14597 C06CVI 23646541 IC50 = 200 nM T14597 C42ONU 23646542 IC50 = 210 nM T14597 C3T8FB 23646543 IC50 > 25000 nM T14597 CVK4Z2 23646544 IC50 = 110 nM T14597 CS31HG 23646545 IC50 = 130 nM T14597 CRQK51 23646546 IC50 = 170 nM T14597 C7O2QA 23646547 IC50 = 9700 nM T14597 C82MEJ 23646548 IC50 = 1400 nM T14597 C08NIK 23646549 IC50 = 2400 nM T14597 CV75ZR 23646550 IC50 = 240 nM T14597 CYWG82 23729145 IC50 > 1000 nM T14597 COV2N4 24179332 IC50 = 13320 nM T14597 C7YG1N 24759534 IC50 = 35000 nM T14597 CAJ4T2 24762205 IC50 > 10000 nM T14597 CCPS81 24764502 IC50 > 35000 nM T14597 C78RNQ 24766872 IC50 = 125 ug.mL-1 T14597 CQ8SY7 24766873 IC50 = 79 ug.mL-1 T14597 C1CGU3 24782374 IC50 = 4 nM T14597 C7DR5J 24782621 IC50 = 843 nM T14597 CFN39G 24782622 IC50 = 2240 nM T14597 CE2Q3V 24786207 IC50 = 960 nM T14597 C43HWQ 24883287 IC50 = 42 nM T14597 C8DA5Q 24883334 IC50 = 18 nM T14597 CB5TP8 24894992 IC50 = 25000 nM T14597 C32SUJ 24894993 IC50 = 36000 nM T14597 CFW40U 24894997 IC50 = 37000 nM T14597 CZ67RA 24897043 IC50 = 2 nM T14597 CVF5W2 24897276 IC50 = 148 nM T14597 CB2EX1 24897277 IC50 = 7 nM T14597 CN9T1Z 24897278 IC50 = 8 nM T14597 C6JA7L 24897279 IC50 = 72 nM T14597 CA5XT2 24897280 IC50 = 39 nM T14597 CN13JF 24899915 IC50 = 8.4 ug.mL-1 T14597 CBWR97 24899916 IC50 = 2.7 ug.mL-1 T14597 C9F2JD 24899917 IC50 > 10 ug.mL-1 T14597 C64MTI 24900160 IC50 > 10 ug.mL-1 T14597 CO2I6Q 24900161 IC50 > 10 ug.mL-1 T14597 C96GPD 24944848 IC50 = 10.6 nM T14597 CNMB03 24944849 IC50 = 12.4 nM T14597 CTCB27 24944850 IC50 = 15 nM T14597 C5PH0N 24944851 IC50 = 20 nM T14597 CK17HZ 24944855 IC50 = 51.6 nM T14597 C0BOJ2 24944856 IC50 = 71.2 nM T14597 CX05SV 24944930 IC50 = 19 nM T14597 CB8EZ0 24944934 IC50 = 38.4 nM T14597 C2CP6T 24944935 IC50 = 38.2 nM T14597 C1NZ8X 24945115 IC50 = 43.5 nM T14597 CF0U4T 24945204 IC50 = 24 nM T14597 C8W3YA 24945368 IC50 = 20.1 nM T14597 C2MYN7 24945689 IC50 = 10.1 nM T14597 C4V9GI 24960018 IC50 > 10000 nM T14597 CIK6V8 25025888 IC50 = 2.5 nM T14597 C0JGL8 25026082 IC50 = 1.6 nM T14597 CHY93R 25026085 IC50 = 6 nM T14597 C3DPS2 25026281 IC50 = 1.7 nM T14597 CHLQ49 25063262 IC50 = 80 nM T14597 CTV54O 25123227 IC50 > 10000 nM T14597 CG3XC9 25124150 IC50 = 72 nM T14597 CO2IR5 25124816 IC50 > 10000 nM T14597 CIG4H0 25178539 IC50 = 7700 nM T14597 CJ3YN8 25195273 IC50 = 6 nM T14597 C8NBA6 25195274 IC50 = 71 nM T14597 C6FGQ1 25206346 IC50 = 1200 nM T14597 C6XQB9 25207010 IC50 = 18 nM T14597 C8LXB1 25218685 IC50 = 186 nM T14597 C3PT8E 25218686 IC50 = 250 nM T14597 CY35SP 25218687 IC50 = 53 nM T14597 CR0FO4 25218688 EC50 = 210 nM T14597 CWNY70 25218689 EC50 = 660 nM T14597 CZ5M3A 25218690 EC50 = 1600 nM T14597 CK9AO6 25218691 EC50 = 1580 nM T14597 CXH7F8 25218692 IC50 = 54 nM T14597 CH2GL3 25218693 EC50 = 147 nM T14597 CQ6MZ0 25242463 IC50 = 100 nM T14597 CM31HJ 25263246 IC50 = 30 nM T14597 CAMY28 25263247 IC50 = 60 nM T14597 C6FB3N 25263248 IC50 = 450 nM T14597 C7P4FS 25263249 IC50 = 260 nM T14597 CV8Y5M 25263250 IC50 = 60 nM T14597 CKG21S 25263251 IC50 = 370 nM T14597 C7I4BG 25263252 IC50 = 180 nM T14597 C9TK3Q 25263253 IC50 = 87 nM T14597 CWE9C6 25263254 IC50 = 60 nM T14597 C9SL4P 25263255 IC50 = 220 nM T14597 C4JQD8 25263256 IC50 = 800 nM T14597 CED02Z 25263257 IC50 = 50 nM T14597 CI79QB 25263258 IC50 = 30 nM T14597 C18VBO 25263259 IC50 = 35 nM T14597 CN89CY 25263260 IC50 = 130 nM T14597 C9JR3E 25263261 IC50 = 85 nM T14597 C0Y9TK 25263263 IC50 = 60 nM T14597 C5I4UQ 25263264 IC50 = 2660 nM T14597 CA0X9R 25263265 IC50 = 180 nM T14597 CW2J5P 25263266 IC50 = 210 nM T14597 CR7JS1 25263267 IC50 = 16 nM T14597 CT60US 25263268 IC50 = 20 nM T14597 C1NAD7 25263269 IC50 = 32 nM T14597 CJI43L 25263270 IC50 = 32 nM T14597 CANP37 25263271 IC50 = 20 nM T14597 CG3OH9 25263272 IC50 = 32 nM T14597 CZ0H9E 25263273 IC50 = 32 nM T14597 CY6HW8 25263274 EC50 = 30 nM T14597 C1WG7S 25263275 EC50 = 50 nM T14597 C6WV8D 25263276 EC50 = 130 nM T14597 CJW7I3 25263277 EC50 = 220 nM T14597 CTO10V 25263278 EC50 = 130 nM T14597 CZ4HN9 25263279 EC50 = 10 nM T14597 C7XEB3 25263280 EC50 = 20 nM T14597 C2ICK6 25263281 EC50 = 120 nM T14597 CZGQ83 25271178 IC50 = 776 nM T14597 CF2LZ7 25271179 IC50 = 1530 nM T14597 CLB28U 25271180 IC50 > 100000 nM T14597 CGHR32 25271181 IC50 > 100000 nM T14597 C3E9XU 25271513 IC50 > 100000 nM T14597 CGBX14 25271514 IC50 = 10000 nM T14597 C76NWM 25271515 IC50 = 10000 nM T14597 C6C4YR 25271516 IC50 > 100000 nM T14597 CUAK50 25271517 IC50 = 776 nM T14597 CIR67H 25271518 IC50 > 100000 nM T14597 CU53WB 42596953 IC50 = 11 nM T14597 C41TLH 42603880 IC50 = 95000 nM T14597 CU9E4P 42629114 IC50 > 10000 nM T14597 CJ5U1X 42639664 IC50 = 4.2 ug.mL-1 T14597 CO42DC 44138048 IC50 > 10000 nM T14597 CL65QV 44138049 IC50 > 10000 nM T14597 C6U2LF 44205208 IC50 = 2.1 nM T14597 CR03OF 44229775 IC50 = 1.6 nM T14597 CEL61X 44229839 IC50 = 0.98 nM T14597 C8DWO1 44229840 IC50 = 3.3 nM T14597 CNM3H2 44229841 IC50 = 6.1 nM T14597 C5BY9T 44279217 IC50 = 21000 nM T14597 C6PO2L 44279342 IC50 = 1860 nM T14597 CO5V3J 44279343 IC50 = 97 nM T14597 C5HE2C 44279364 IC50 = 1100 nM T14597 C5ERW7 44279376 IC50 = 1300 nM T14597 C5AWJ0 44279421 IC50 = 27000 nM T14597 C9C2KB 44279443 IC50 = 290 nM T14597 CI7R0U 44279655 IC50 = 350 nM T14597 C21LXN 44279656 IC50 = 3100 nM T14597 CLKP81 44307006 IC50 = 6600 nM T14597 CVFL96 44307008 IC50 = 3800 nM T14597 CSY8A3 44321301 IC50 = 19000 nM T14597 CCG2M5 44321317 IC50 = 8200 nM T14597 CY9ED1 44321395 IC50 = 15200 nM T14597 C5U1CR 44321686 IC50 > 10000 nM T14597 CETY53 44321717 IC50 > 100000 nM T14597 CV60ME 44321734 IC50 > 50000 nM T14597 CGHA16 44325116 IC50 = 117 nM T14597 CW42OA 44345288 IC50 = 8709.64 nM T14597 C0A6IM 44345309 IC50 = 10000 nM T14597 CO9U4D 44345316 IC50 = 707.95 nM T14597 C57GUL 44345336 IC50 = 446.68 nM T14597 C09YJV 44345337 IC50 = 112201.85 nM T14597 CL73FP 44345342 IC50 = 17378.01 nM T14597 CI02JL 44345396 IC50 = 15135.61 nM T14597 CHE2P1 44345431 IC50 = 10000 nM T14597 CRQ76V 44345433 IC50 = 1023.29 nM T14597 CJB1C4 44345439 IC50 = 3311.31 nM T14597 CVZ05R 44345469 IC50 = 2511.89 nM T14597 C06AQN 44345644 IC50 = 6165.95 nM T14597 CD62QG 44345647 IC50 = 1513.56 nM T14597 C2ESL8 44345648 IC50 = 1659.59 nM T14597 CK4U5B 44361553 IC50 = 4570.88 nM T14597 CM56JY 44361640 IC50 = 2884.03 nM T14597 CT2R7Z 44361668 IC50 = 1995.26 nM T14597 C5RZI9 44361703 IC50 = 20892.96 nM T14597 C04PXM 44361706 IC50 = 15848.93 nM T14597 C7X2IR 44361708 IC50 = 91201.08 nM T14597 C1NRF6 44361710 IC50 = 4570.88 nM T14597 C10VDK 44371971 IC50 = 380 nM T14597 C2GRI5 44372004 IC50 = 110 nM T14597 C9NYG0 44372005 IC50 = 60 nM T14597 CFM6C8 44372022 IC50 = 14 nM T14597 CCGX21 44372180 IC50 = 200 nM T14597 C6L4CX 44372197 IC50 = 1500 nM T14597 CSA68M 44372283 IC50 = 15000 nM T14597 C87MAJ 44388483 IC50 = 3900 nM T14597 CB7QM3 44388486 IC50 = 171 nM T14597 C6WDG3 44388487 IC50 = 1100 nM T14597 C3YM9F 44388494 IC50 = 227 nM T14597 CN4L2V 44388499 IC50 = 412 nM T14597 CUA90G 44388501 IC50 = 13000 nM T14597 C4GV1S 44399994 IC50 = 310000 nM T14597 CH9NR8 44403081 IC50 = 7200 nM T14597 C0AR9C 44403420 IC50 = 5 nM T14597 CGQ26K 44403425 IC50 = 1100 nM T14597 CRV6B4 44403429 IC50 = 24 nM T14597 CTY5K7 44403435 IC50 = 70 nM T14597 C47XFZ 44403436 IC50 = 24 nM T14597 C7HD4Q 44410411 IC50 = 21000 nM T14597 CED5S6 44410414 IC50 = 3800 nM T14597 C0A7XB 44410560 IC50 = 91 nM T14597 C5WKG0 44410574 IC50 = 1820 nM T14597 CDQ4S6 44410648 IC50 = 66 nM T14597 C4OJ1S 44410700 IC50 = 45 nM T14597 CIY53K 44410704 IC50 = 32 nM T14597 CPH17L 44410710 IC50 = 32 nM T14597 C2J1KU 44410716 IC50 = 29 nM T14597 C0XJC3 44412177 IC50 = 11800 nM T14597 C5QD2S 44412181 IC50 = 23030 nM T14597 CRH3Y6 44412244 IC50 = 11080 nM T14597 C16IVC 44416188 IC50 = 38 nM T14597 COFI73 44416243 IC50 = 35 nM T14597 CS8U4Y 44416288 IC50 = 30 nM T14597 CVA3S4 44416289 IC50 = 26 nM T14597 CY13SQ 44418977 IC50 = 560 nM T14597 CN15DI 44426255 IC50 > 10000 nM T14597 CTO06X 44426256 IC50 > 10000 nM T14597 CJC0Q4 44426257 IC50 > 10000 nM T14597 C3ZHQ5 44426258 IC50 = 51 nM T14597 C7D0WF 44426259 IC50 = 75 nM T14597 CCW18G 44426260 IC50 = 16 nM T14597 CA09HO 44426261 IC50 > 10000 nM T14597 CU04XF 44426262 IC50 = 550 nM T14597 CEJ9W5 44426263 IC50 = 76 nM T14597 C7EW8J 44426264 IC50 > 10000 nM T14597 C7TI3M 44426265 IC50 > 10000 nM T14597 C07GXY 44426266 IC50 = 140 nM T14597 C8FZ0A 44426267 IC50 = 160 nM T14597 C4YE5V 44426268 IC50 = 18 nM T14597 CPYM43 44426269 IC50 = 130 nM T14597 CE69XZ 44426270 IC50 > 10000 nM T14597 CS1FQ0 44426271 IC50 > 10000 nM T14597 COE84X 44426272 IC50 > 10000 nM T14597 C23ZTG 44426273 IC50 > 10000 nM T14597 C4OI5J 44426274 IC50 = 140 nM T14597 CNS0Q7 44426275 IC50 = 260 nM T14597 C5MF1L 44426276 IC50 = 19 nM T14597 C3LV1P 44426277 IC50 = 34 nM T14597 C9QI8R 44426278 IC50 < 10 nM T14597 CTYU67 44426279 IC50 < 10 nM T14597 CN9I7M 44426280 IC50 = 230 nM T14597 CNJV25 44426281 IC50 = 27 nM T14597 C74NTR 44426282 IC50 = 55 nM T14597 CZ5Y8R 44426283 IC50 = 25 nM T14597 CPD21M 44426284 IC50 = 530 nM T14597 CU1GZ0 44426285 IC50 = 44 nM T14597 CD1V6I 44426286 IC50 = 30 nM T14597 C0CW2T 44426287 IC50 = 280 nM T14597 CP5R4Z 44426288 IC50 < 10 nM T14597 CT28VH 44426289 IC50 < 10 nM T14597 CH3Z2D 44426290 IC50 = 21 nM T14597 CF8G2B 44426291 IC50 = 15 nM T14597 C7BZ0K 44430019 IC50 = 88 nM T14597 CJ1U9R 44430027 IC50 > 1000 nM T14597 COBA27 44430030 IC50 = 310 nM T14597 C8WJV9 44430032 IC50 = 120 nM T14597 C9UYP5 44430034 IC50 = 16 nM T14597 CQ67VA 44430037 IC50 = 170 nM T14597 CW58IO 44430039 IC50 = 74 nM T14597 CWC6X5 44437843 IC50 = 36500 nM T14597 CR0YC3 44437845 IC50 > 50000 nM T14597 CRED62 44437846 IC50 > 50000 nM T14597 CWVI75 44437847 IC50 > 50000 nM T14597 C2LTG9 44437848 IC50 = 31600 nM T14597 C03YUM 44437849 IC50 = 16600 nM T14597 CX09ZA 44440812 IC50 > 1000 nM T14597 C36FXV 44440815 IC50 = 110 nM T14597 CF5UR8 44440816 IC50 = 310 nM T14597 C87FRB 44440817 IC50 = 250 nM T14597 CNCU91 44440820 IC50 = 420 nM T14597 CL1N3P 44440821 IC50 = 420 nM T14597 C85SOF 44440823 IC50 = 18 nM T14597 C8GHB0 44440824 IC50 = 280 nM T14597 C74ONA 44440826 IC50 = 110 nM T14597 CNU0P1 44440830 IC50 = 120 nM T14597 CU72VL 44440831 IC50 = 170 nM T14597 CNY07A 44440833 IC50 = 60 nM T14597 CZ4G2C 44440835 IC50 = 590 nM T14597 C85HCV 44440836 IC50 = 140 nM T14597 CO6DP3 44440837 IC50 = 560 nM T14597 C4Y1TD 44440839 IC50 = 380 nM T14597 CWC9V6 44440840 IC50 = 410 nM T14597 CIF14K 44440841 IC50 = 130 nM T14597 CJ23DP 44440842 IC50 = 850 nM T14597 CO8WZ7 44440843 IC50 = 41 nM T14597 CJL0G8 44440844 IC50 = 510 nM T14597 CA75PM 44440874 IC50 = 250 nM T14597 CAM78I 44441000 IC50 = 52 nM T14597 C6ZEJ5 44441012 IC50 = 170 nM T14597 C3MW6G 44441013 IC50 = 43 nM T14597 C3AZF8 44441014 IC50 = 35 nM T14597 CJC06N 44441015 IC50 = 34 nM T14597 CWJ1U3 44441016 IC50 = 190 nM T14597 C2IL0Y 44441017 IC50 = 13 nM T14597 CMW7T5 44442025 IC50 < 2 nM T14597 C3U1GC 44442026 IC50 = 19 nM T14597 C9J2FM 44442027 IC50 < 2 nM T14597 CU7N0D 44442028 IC50 = 22 nM T14597 CF4DL2 44446843 IC50 = 358 nM T14597 CT9R7H 44448969 IC50 = 4123 nM T14597 C9RV4Q 44448995 IC50 = 5220 nM T14597 CUB12D 44449577 IC50 = 500 nM T14597 C7HIM2 44452543 IC50 > 500 nM T14597 CZ9H4D 44452544 IC50 > 500 nM T14597 CQ1M7K 44455194 IC50 < 1 nM T14597 C86DQE 44455195 IC50 = 4 nM T14597 C20ISD 44455293 IC50 = 613 nM T14597 CUN90T 44455330 IC50 = 5 nM T14597 C4Z0WX 44455645 IC50 = 30 nM T14597 C75RIH 44455672 IC50 = 120 nM T14597 C7LJ2U 44455701 IC50 = 23 nM T14597 CIQ3O8 44455702 IC50 = 27 nM T14597 CY5PB6 44455730 IC50 = 22 nM T14597 CBID06 44455782 IC50 = 31 nM T14597 CAS03E 44481081 IC50 = 6490 nM T14597 C4TF5E 44481332 IC50 = 6730 nM T14597 CDFI53 44528870 IC50 = 246 nM T14597 CI8X2C 44528924 IC50 = 76 nM T14597 C9ZU2D 44528930 IC50 = 153 nM T14597 CXR98Y 44528960 IC50 = 68 nM T14597 CFP97X 44532811 IC50 = 31 nM T14597 C1A4XG 44562420 IC50 = 146 nM T14597 C3UV2W 44562431 IC50 = 5700 nM T14597 CC62JT 44564704 IC50 = 120 nM T14597 CC7E4K 44564705 IC50 > 10000 nM T14597 C42ZEW 44564706 IC50 = 1100 nM T14597 C53MCK 44564747 IC50 > 10000 nM T14597 CDI31F 44564748 IC50 > 10000 nM T14597 CA17NT 44564749 IC50 > 10000 nM T14597 CSO9F8 44564751 IC50 > 10000 nM T14597 CM50GS 44564788 IC50 > 10000 nM T14597 C3Q0DX 44564789 IC50 = 3100 nM T14597 CP40XB 44564790 IC50 = 1600 nM T14597 C35NTB 44564791 IC50 > 10000 nM T14597 CJY83G 44564817 IC50 > 10000 nM T14597 CF2D1K 44564819 IC50 > 10000 nM T14597 C3CQ9K 44564820 IC50 > 10000 nM T14597 CI8V2L 44564821 IC50 > 10000 nM T14597 C9PO7J 44564860 IC50 > 10000 nM T14597 C16FJW 44564861 IC50 > 10000 nM T14597 CRX0M5 44571414 IC50 = 299 nM T14597 C9KY2N 44571415 IC50 = 203 nM T14597 CT92ZI 44571431 IC50 = 709 nM T14597 C0W9NE 44571432 IC50 = 86 nM T14597 CKY57M 44571433 IC50 = 113 nM T14597 C2RQ3H 44571434 IC50 = 113 nM T14597 CUCI91 44571435 IC50 = 14 nM T14597 C7LVG6 44571436 IC50 = 898 nM T14597 CIU14N 44571437 IC50 = 111 nM T14597 CLP71D 44571448 IC50 = 146 nM T14597 CEIK76 44571449 IC50 = 250 nM T14597 CFNT92 44571450 IC50 = 122 nM T14597 CIB7R5 44571451 IC50 = 68 nM T14597 CK6L2W 44571452 IC50 = 121 nM T14597 CI1PL5 44571453 IC50 = 43 nM T14597 CZ0ID1 44571454 IC50 = 95 nM T14597 CWFB42 44571820 IC50 = 54 nM T14597 C5TE0I 44575454 IC50 = 8.5 ug.mL-1 T14597 C1ARI6 44575455 IC50 = 6 ug.mL-1 T14597 C9XIA1 44580891 IC50 = 54 nM T14597 CZC2R9 44580892 IC50 = 110 nM T14597 CYSF35 44580915 IC50 = 88 nM T14597 CP81ZN 44580916 IC50 = 38 nM T14597 CQL7G0 44580917 IC50 = 120 nM T14597 C8LK3H 44580918 IC50 = 11 nM T14597 C5H1XE 44580949 IC50 = 98 nM T14597 C2I8SC 44580950 IC50 = 40 nM T14597 CK9NC7 44580951 IC50 = 90 nM T14597 CO6A7L 44580971 IC50 = 135 nM T14597 CHSR02 44581016 IC50 = 78 nM T14597 C06LHO 44581017 IC50 = 87 nM T14597 C2Z4HB 44583600 IC50 = 137 nM T14597 CD4Q8C 44583601 IC50 = 28 nM T14597 CD2AQ7 44583620 IC50 = 194 nM T14597 CLZ6X5 44583621 IC50 = 102 nM T14597 C5HA4P 44583622 IC50 = 470 nM T14597 C7PR8I 44583623 IC50 = 100 nM T14597 CDRC42 44583654 IC50 = 18 nM T14597 C5HEX6 44583655 IC50 = 170 nM T14597 CM79HD 44583656 IC50 = 67 nM T14597 CF6Z2N 44585507 IC50 = 19 nM T14597 CRL65K 44585537 IC50 = 13 nM T14597 C3KUW4 44585573 IC50 = 733 nM T14597 CUA35G 44585574 IC50 = 1700 nM T14597 C6CJ4Y 44585594 IC50 = 5300 nM T14597 CQV6W9 44586019 IC50 = 8 nM T14597 CTHK89 44587526 IC50 = 118 nM T14597 C7BP3R 44587569 IC50 = 8 nM T14597 C2TAB7 44593674 IC50 = 8 ug.mL-1 T14597 CM0I4J 45101511 IC50 = 27.5 nM T14597 CXR3J0 45140149 IC50 = 76.5 nM T14597 C42EAO 45140150 IC50 = 24.2 nM T14597 CQ0WZ2 45140151 IC50 > 2000 nM T14597 CCLE50 45140153 IC50 = 225.2 nM T14597 C4QVP3 45140347 IC50 = 295.4 nM T14597 CR8GN7 45140348 IC50 > 2000 nM T14597 C6K1JW 45140349 IC50 = 27.8 nM T14597 C82WLQ 45140350 IC50 = 175 nM T14597 CR4C9A 45140351 IC50 = 556.9 nM T14597 C4UM6Y 45273507 IC50 > 10000 nM T14597 C6E2SC 45482700 IC50 > 10000 nM T14597 CZXH74 45482750 IC50 > 10000 nM T14597 CB6X7D 45483674 IC50 = 18 nM T14597 CCMU48 45483675 IC50 = 22 nM T14597 C9PE3R 45483677 IC50 = 20 nM T14597 CF9SL7 45483685 IC50 = 37 nM T14597 CE7J8I 45483687 IC50 = 23 nM T14597 CULV14 45483689 IC50 = 29 nM T14597 C2V0QA 45483691 IC50 = 44 nM T14597 CFN61Z 45483693 IC50 = 28 nM T14597 CET9K4 45483694 IC50 = 30 nM T14597 CJ1XL4 45483695 IC50 = 18 nM T14597 CO0U2K 45483696 IC50 = 21 nM T14597 CKSM90 45483699 IC50 = 77 nM T14597 CZS39O 45487302 IC50 = 29 nM T14597 C4ZWY7 45487310 IC50 = 44.5 nM T14597 C9SV0H 45487311 IC50 = 3.8 nM T14597 C6GCM7 45487332 IC50 = 4.3 nM T14597 CCF05Q 45487333 IC50 = 5.6 nM T14597 C23NRD 45487334 IC50 = 50.5 nM T14597 CY09ZU 45487335 IC50 = 7.3 nM T14597 CQHJ85 45487342 IC50 = 15.5 nM T14597 C3ZLN1 45487343 IC50 = 10 nM T14597 CI6DW2 45487357 IC50 = 8.5 nM T14597 COX40Y 45487358 IC50 = 42 nM T14597 CF1T7M 45487359 IC50 = 4.4 nM T14597 CRXI29 45487373 IC50 = 3.8 nM T14597 CYL32E 45487376 IC50 = 11 nM T14597 CO5P9I 45487386 IC50 = 28 nM T14597 CS9Y8G 45487387 IC50 = 70 nM T14597 CAN4J2 45487388 IC50 = 162 nM T14597 CWLC18 45487393 IC50 = 11.5 nM T14597 CO9NJ2 45487398 IC50 = 5.6 nM T14597 CDN5Q6 45487399 IC50 = 52 nM T14597 CI4KJ5 45487400 IC50 = 8.1 nM T14597 C49HOI 45487401 IC50 = 31 nM T14597 CBK43U 45487402 IC50 = 30 nM T14597 C5VC7I 46200951 IC50 = 350 nM T14597 C5G7SV 46207008 IC50 = 9950 nM T14597 CA3N9W 46207009 IC50 = 2580 nM T14597 C4K9MS 46207010 IC50 = 3890 nM T14597 CAE1M9 46207011 IC50 = 12870 nM T14597 C2F4HI 46207012 IC50 = 15390 nM T14597 C7CID4 46207014 IC50 = 46100 nM T14597 C9CER0 46207015 IC50 > 50000 nM T14597 CPI6S1 46207036 IC50 = 39640 nM T14597 C3F6SM 46207037 IC50 > 50000 nM T14597 C10WUT 46207039 IC50 = 48350 nM T14597 CPXZ65 46207040 IC50 = 30060 nM T14597 C30QNX 46207041 IC50 = 22750 nM T14597 CDN84U 46207042 IC50 = 350 nM T14597 CV1P0R 46207043 IC50 = 25870 nM T14597 C41RBD 46207062 IC50 = 27190 nM T14597 CBQS73 46207441 IC50 = 2320 nM T14597 C1WS6M 46207442 IC50 = 3330 nM T14597 CUA97D 46209401 IC50 > 10000 nM T14597 CY3HW5 46224684 IC50 > 10000 nM T14597 C8YPN0 46225596 IC50 = 3600 nM T14597 C34JTS 46225597 IC50 > 10000 nM T14597 CGD73B 46225598 IC50 > 10000 nM T14597 C3E0PU 46225599 IC50 > 10000 nM T14597 CRDY89 46225610 IC50 = 38 nM T14597 C0JMT8 46225611 IC50 = 130 nM T14597 CF0D5J 46225612 IC50 = 100 nM T14597 CFVO38 46225632 IC50 > 10000 nM T14597 CLZ1O6 46225634 IC50 = 2400 nM T14597 C07VDX 46225635 IC50 = 2200 nM T14597 CT70DX 46225640 IC50 = 32 nM T14597 CJUF68 46225641 IC50 = 180 nM T14597 C6AJ5N 46225647 IC50 = 6950 nM T14597 C2WCV1 46225648 IC50 > 10000 nM T14597 CBS96A 46225649 IC50 > 10000 nM T14597 C38BFC 46225657 IC50 = 5 nM T14597 CD0A6F 46225658 IC50 = 5900 nM T14597 C1B3KS 46225663 IC50 = 300 nM T14597 CU46XI 46225664 IC50 = 2300 nM T14597 CO3HS2 46225665 IC50 > 10000 nM T14597 C2UV1S 46225666 IC50 > 10000 nM T14597 CX5B1G 46225667 IC50 > 10000 nM T14597 CM14FH 46225680 IC50 = 2300 nM T14597 CQS96E 46225681 IC50 > 10000 nM T14597 CJIK35 46225682 IC50 = 47 nM T14597 C8S4QA 46225688 IC50 = 490 nM T14597 CYBD14 46229355 IC50 = 3450 nM T14597 C7XEG1 46229356 IC50 = 5170 nM T14597 CO0DJ5 46229377 IC50 = 38230 nM T14597 C5Y1PT 46229378 IC50 = 9640 nM T14597 CE25DB 46229379 IC50 = 12420 nM T14597 CT70VJ 46229380 IC50 > 50000 nM T14597 CT15NR 46229381 IC50 = 2270 nM T14597 CG14AQ 46229405 IC50 = 2660 nM T14597 CK7BT5 46229406 IC50 = 18430 nM T14597 CKN40P 46229407 IC50 = 2210 nM T14597 CKL7Z5 46229408 IC50 = 4530 nM T14597 C3IS6A 46229409 IC50 = 16120 nM T14597 CEK82A 46229459 IC50 > 50000 nM T14597 C3N0HQ 46229460 IC50 > 50000 nM T14597 CAO23J 46229461 IC50 > 50000 nM T14597 CJ3FW1 46229462 IC50 > 50000 nM T14597 CI6RL4 46229463 IC50 > 50000 nM T14597 CQ8K2T 46229464 IC50 > 50000 nM T14597 C2SF0M 46229498 IC50 = 1410 nM T14597 CY4K7S 46229499 IC50 = 1870 nM T14597 C9YBX1 46229500 IC50 = 15660 nM T14597 CF4P3E 46229516 IC50 = 37820 nM T14597 CI1X8G 46229517 IC50 = 660 nM T14597 CH91IA 46229518 IC50 = 7130 nM T14597 CW40RS 46229519 IC50 = 1230 nM T14597 CS3OP4 46229535 IC50 = 2240 nM T14597 C7UOQ9 46229536 IC50 = 9470 nM T14597 C4MA6T 46229537 IC50 = 32540 nM T14597 CUSX60 46229538 IC50 = 39510 nM T14597 CAKH92 46229539 IC50 > 50000 nM T14597 CLOQ02 46229565 IC50 = 39780 nM T14597 CWD64Q 46229566 IC50 > 50000 nM T14597 CJ4NH6 46229567 IC50 > 50000 nM T14597 CGMY03 46229773 IC50 = 410 nM T14597 C5D0OS 46229856 IC50 = 44510 nM T14597 CYZV41 46231219 IC50 > 8480 nM T14597 C7J5UP 46231220 IC50 = 15180 nM T14597 CC96GZ 46231221 IC50 = 13316 nM T14597 CS8P3R 46233390 IC50 = 478.2 nM T14597 CZD79U 46831432 IC50 = 970 nM T14597 CNWU53 46831433 IC50 = 980 nM T14597 CD3TK2 46842884 IC50 = 2770 nM T14597 C39RVL 46846074 IC50 = 2290 nM T14597 CE3WH9 46865125 IC50 = 0.5 nM T14597 C45LYT 46865445 IC50 = 26.1 nM T14597 CCBE34 46865992 IC50 = 4.3 nM T14597 C1XEY4 46866615 IC50 = 10.6 nM T14597 CF6K3E 46866616 IC50 = 2.9 nM T14597 CLS29B 46872626 IC50 > 10000 nM T14597 C2MCT8 46879471 IC50 > 5000 nM T14597 C6M0JK 46879472 IC50 = 934 nM T14597 CGV58U 46879473 IC50 = 3840 nM T14597 C8GD2E 46879474 IC50 = 620 nM T14597 CF4OY7 46881850 IC50 = 54 nM T14597 CEKX49 46881918 IC50 = 54 nM T14597 CAB87H 46886244 IC50 > 12500 nM T14597 C92HEB 46886245 IC50 = 240 nM T14597 C5WFQ8 46886310 IC50 = 35 nM T14597 C7S8RG 46886311 IC50 = 6.3 nM T14597 CO13IV 46886312 IC50 = 6000 nM T14597 C70PZE 46886313 IC50 = 4.8 nM T14597 CE8HR2 46886314 IC50 = 86 nM T14597 CG5KO9 46886315 IC50 = 1400 nM T14597 CIFR42 46886316 IC50 = 1300 nM T14597 CH5DC2 46886317 IC50 = 170 nM T14597 C2WKO4 46886318 IC50 = 170 nM T14597 CMVZ46 46886319 IC50 = 370 nM T14597 CW19TR 46886320 IC50 = 86 nM T14597 CJR01I 46886321 IC50 = 14 nM T14597 CL50ZE 46886322 IC50 = 7.2 nM T14597 C2O8RZ 46886323 IC50 = 73 nM T14597 CN30BX 46886324 IC50 = 160 nM T14597 CC7MG8 46886325 IC50 = 170 nM T14597 C0L1EW 46886326 IC50 = 150 nM T14597 C3T6YO 46886327 IC50 = 120 nM T14597 C0WYM1 46898022 IC50 = 10000 nM T14597 C70IVU 46906826 IC50 = 1320 nM T14597 CRI1Q8 46912936 IC50 = 2150 nM T14597 CPR6O9 47108694 IC50 = 13070 nM T14597 CM24GY 47108695 IC50 = 8410 nM T14597 CF9ZH7 47108713 IC50 = 19050 nM T14597 C4FJ0Y 49798860 IC50 = 5030 nM T14597 CBX8W0 49798861 IC50 = 9240 nM T14597 C8AWO3 49799240 IC50 = 6580 nM T14597 COD7X8 49799764 IC50 = 4650 nM T14597 C3PNH8 49799765 IC50 = 9650 nM T14597 CO89EH 49799766 IC50 = 14320 nM T14597 C4MYV3 49799767 IC50 = 9970 nM T14597 CK92JP 49799768 IC50 = 3460 nM T14597 CY32VC 49799770 IC50 = 40000 nM T14597 C21GOI 49799777 IC50 = 5840 nM T14597 C7QR3M 49799778 IC50 = 4770 nM T14597 CVEG83 49799781 IC50 = 41260 nM T14597 C6X5MK 49799782 IC50 = 36450 nM T14597 C2GXI7 49799783 IC50 = 44850 nM T14597 C1NI4A 49799785 IC50 > 50000 nM T14597 C3VQ9Z 49799786 IC50 = 19340 nM T14597 CAL42P 49799787 IC50 = 16750 nM T14597 C49XCZ 49799788 IC50 = 18820 nM T14597 C5ME3S 49806721 IC50 > 50000 nM T14597 CE7D2J 49855568 IC50 = 4.1 nM T14597 CFD9P3 49855569 IC50 = 3.5 nM T14597 C1AU5N 49855758 IC50 = 12 nM T14597 CIFK93 49855759 IC50 = 5.7 nM T14597 CK48OJ 49855760 IC50 = 4.9 nM T14597 CZI3M1 49855761 IC50 = 8.7 nM T14597 CRPZ58 49855949 IC50 = 14 nM T14597 CTU0K3 49855950 IC50 = 15 nM T14597 CF85NL 49855951 IC50 = 4.7 nM T14597 CF7YS9 49855952 IC50 = 2 nM T14597 CJU38G 49855953 IC50 = 3.5 nM T14597 CS9G6E 50997096 IC50 > 10000 nM T14597 CM42BY 51000510 Ki > 1000000 nM T14597 C49ZVC 51346878 IC50 = 440 nM T14597 CJ4L1K 51346887 IC50 = 190 nM T14597 CH1TU2 51346888 IC50 = 19 nM T14597 C2ZTN3 52941514 IC50 = 16 nM T14597 C8XN0Y 52941515 IC50 = 5230 nM T14597 CT37AH 52942747 IC50 = 478 nM T14597 CA51LB 52943781 IC50 = 14.5 nM T14597 CD5YH8 52946371 IC50 = 9.8 nM T14597 CGA62C 52946372 IC50 = 13.8 nM T14597 C09UQW 52946470 IC50 = 15.4 nM T14597 CIC58E 52946503 IC50 = 334 nM T14597 CQ87LD 52946569 IC50 = 215 nM T14597 CQ0V4I 52947602 IC50 = 21.5 nM T14597 CYQ4L3 52947603 IC50 = 29 nM T14597 CTY9Z8 52948817 IC50 = 21.5 nM T14597 CPAM54 52950015 IC50 > 62500 nM T14597 C0M2SG 52950017 IC50 = 15.1 nM T14597 CJ61BU 53317172 IC50 > 100000 nM T14597 C89QOE 53317173 IC50 = 140 nM T14597 C50BWT 53317174 IC50 = 3750 nM T14597 C39KUD 53317175 IC50 = 70 nM T14597 CBHT02 53318117 IC50 = 360 nM T14597 CX1V9L 53318118 IC50 = 20 nM T14597 C90MNQ 53318457 IC50 = 6500 nM T14597 C2X8OF 53318458 IC50 = 78 nM T14597 CK59QY 53318459 IC50 = 810 nM T14597 CRBE56 53319790 IC50 = 150 nM T14597 CSC61X 53320059 IC50 = 318 nM T14597 CX65KS 53321087 IC50 > 100000 nM T14597 CX7S8I 53322057 IC50 = 880 nM T14597 CSY76U 53322058 IC50 = 70 nM T14597 C7Y3ZR 53322413 IC50 = 2900 nM T14597 CR12OB 53322414 IC50 = 102 nM T14597 CR4K7J 53322690 IC50 = 1800 nM T14597 CT1BN7 53324027 IC50 > 100000 nM T14597 C43BZJ 53324200 IC50 = 65000 nM T14597 C2W9OA 53324451 IC50 > 10000 nM T14597 CG18XC 53325046 IC50 = 6300 nM T14597 CD91UQ 53325047 IC50 = 36000 nM T14597 C5C1UW 53325048 IC50 = 740 nM T14597 CRT07X 53325049 IC50 = 81 nM T14597 C69AUF 53325050 IC50 = 95 nM T14597 CN1X9I 53325551 IC50 = 71 nM T14597 C36OQR 53325588 IC50 > 1000 nM T14597 C07PMQ 53326342 IC50 = 5380 nM T14597 CNPM14 53341082 IC50 = 22.4 nM T14597 CM7P3W 53357328 IC50 > 50000 nM T14597 CBK9Q6 53357848 IC50 > 10000 nM T14597 CUZH35 54754343 IC50 = 1530 nM T14597 C1XS2J 54760383 IC50 = 60 nM T14597 CQ17GA 56640518 IC50 = 1 nM T14597 CG20VK 56640520 IC50 = 3.6 nM T14597 CZ9C8M 56640588 IC50 = 15.5 nM T14597 CH0D7P 56640590 IC50 = 3.4 nM T14597 C2PYI1 56659875 IC50 = 13560 nM T14597 CT5NK2 56659876 IC50 = 20330 nM T14597 C2MW9D 56659883 IC50 = 23460 nM T14597 CD67RU 56663333 IC50 = 15570 nM T14597 CCR3V9 56663334 IC50 = 25030 nM T14597 C7NF0U 56666765 IC50 = 4210 nM T14597 C9LPB6 56666766 IC50 = 23450 nM T14597 C4S9ID 56666767 IC50 = 37930 nM T14597 C4L2QB 56670196 IC50 = 4760 nM T14597 CIPW74 56670197 IC50 = 3410 nM T14597 CSNH68 56670198 IC50 = 18940 nM T14597 C97LHS 56670199 IC50 = 19830 nM T14597 C6W7BR 56670200 IC50 > 50000 nM T14597 CRXF95 56673721 IC50 = 7560 nM T14597 CG9N7C 56673722 IC50 = 8180 nM T14597 CFAT97 56673723 IC50 = 29070 nM T14597 CXP5G4 56677027 IC50 = 16260 nM T14597 C6ME8I 56680356 IC50 = 3590 nM T14597 CNLI27 56680357 IC50 = 10530 nM T14597 CN28KJ 56680358 IC50 = 11050 nM T14597 COK71Z 56683687 IC50 = 7020 nM T14597 CQ8Z1X 56683695 IC50 = 26330 nM T14597 C5GM0Z 56683696 IC50 = 27890 nM T14597 CNL0A1 56683697 IC50 = 20450 nM T14597 CP7M1A 56683698 IC50 = 27380 nM T14597 CR50TJ 56835147 IC50 > 10000 nM T14597 CI5ZJ7 56835161 IC50 = 62 nM T14597 CH42FN 56849555 IC50 = 22 nM T14597 C7EOC6 56849556 IC50 = 60 nM T14597 C41DXG 56849558 IC50 = 3.3 nM T14597 C7EC6L 56849560 IC50 = 11 nM T14597 CSXO65 56849562 IC50 = 17 nM T14597 CM9X2J 56849563 IC50 = 4.1 nM T14597 CJRC62 56849701 IC50 = 12 nM T14597 C70VDK 56849702 IC50 = 29 nM T14597 C57FAZ 56849703 IC50 = 2.1 nM T14597 C3BOK4 56849704 IC50 = 8.4 nM T14597 C5XR7P 56849846 IC50 = 4.3 nM T14597 CWX3F4 56849847 IC50 = 5.7 nM T14597 C8D6BW 56849848 IC50 = 15 nM T14597 C62JNG 56849850 IC50 = 2.8 nM T14597 CR49PX 56850806 IC50 = 15 nM T14597 CRT19B 56850930 IC50 = 7.7 nM T14597 CL4A9X 56851051 IC50 = 9.4 nM T14597 C1C0XN 56851052 IC50 = 12 nM T14597 C3HXG6 56851053 IC50 = 12 nM T14597 C6U4YJ 56851166 IC50 = 12 nM T14597 CNA4S2 56851288 IC50 = 19 nM T14597 C7VDW1 56851290 IC50 = 16 nM T14597 C0HNY8 56851427 IC50 = 9.3 nM T14597 C86DBO 56851428 IC50 = 20 nM T14597 C05DWH 56851429 IC50 = 11 nM T14597 C4I0GV 56851430 IC50 = 8.3 nM T14597 CITG07 56851431 IC50 = 8 nM T14597 C1JY4V 56851432 IC50 = 8.2 nM T14597 C2YRQ5 56851433 IC50 = 720 nM T14597 C90MDR 56851588 IC50 = 120 nM T14597 C9NGK2 56851589 IC50 = 30 nM T14597 CZ8UE4 56851590 IC50 = 55 nM T14597 CR0FI9 56851591 IC50 = 41 nM T14597 CYZL68 56851592 IC50 = 4.6 nM T14597 C2JV6S 56851593 IC50 = 26 nM T14597 C6S5PN 56851594 IC50 = 13 nM T14597 CQ2U4F 56949987 IC50 = 29 nM T14597 C86USY 56950114 IC50 = 42 nM T14597 CCTI03 56950115 IC50 = 38 nM T14597 C5K3PV 56950116 IC50 = 79 nM T14597 C8O4DU 57390197 IC50 = 559 nM T14597 C0E5UQ 57390198 IC50 = 135 nM T14597 CLB4Q9 57390199 IC50 = 196 nM T14597 C04YLM 57390200 IC50 > 10000 nM T14597 COC5Y3 57390776 IC50 = 41 nM T14597 C20OVM 57390777 IC50 = 30 nM T14597 C80RNH 57391987 IC50 = 3740 nM T14597 C8U9EO 57391988 IC50 = 834 nM T14597 CHS82P 57392588 IC50 = 41 nM T14597 CZBJ71 57392589 IC50 = 140 nM T14597 CH12GK 57392590 IC50 = 110 nM T14597 CY2XK0 57392591 IC50 = 120 nM T14597 CTB8R9 57394107 IC50 = 1293 nM T14597 C9CO0F 57395424 IC50 > 10000 nM T14597 CM18WP 57396070 IC50 = 130 nM T14597 C6NC2K 57397269 IC50 = 219 nM T14597 C87OHQ 57397677 IC50 > 10000 nM T14597 CO24DL 57397871 IC50 = 220 nM T14597 C5D1MK 57397872 IC50 = 180 nM T14597 CG9E5X 57399346 IC50 = 1234 nM T14597 CO34ZJ 57400426 IC50 = 73 nM T14597 CC3U6B 57400808 IC50 > 40000 nM T14597 CQ5MB9 57401285 IC50 = 750 nM T14597 CMP96A 57401286 IC50 = 86 nM T14597 CKVJ46 57402440 IC50 = 2421 nM T14597 CD0W6U 57402866 IC50 = 2138 nM T14597 CT7M3G 57413593 IC50 = 2 nM T14597 CM9OF3 57413596 IC50 = 2.2 nM T14597 C1RS3Y 57415414 IC50 = 1.3 nM T14597 C80BOQ 57415415 IC50 = 18 nM T14597 CSV93M 57415416 IC50 = 28 nM T14597 C3H6UJ 57415417 IC50 = 130 nM T14597 CW5IS7 57415418 IC50 = 150 nM T14597 C1DS4B 57415535 IC50 = 2.5 nM T14597 C0W8LA 57415536 IC50 = 1.5 nM T14597 CRB83E 57415537 IC50 = 2.1 nM T14597 CI5U3G 57496699 IC50 = 11 nM T14597 CZ35GD 57496700 IC50 = 2.3 nM T14597 CWVJ06 57597166 IC50 = 6.3 nM T14597 CVS51B 57597223 IC50 = 11 nM T14597 C0QUZ4 57597316 IC50 = 17 nM T14597 CD0M7X 57597387 IC50 = 7.1 nM T14597 C4V7FY 58191950 IC50 = 2900 nM T14597 CPCA29 58191961 IC50 = 3400 nM T14597 C7HF1L 58191965 IC50 = 66 nM T14597 C8LWY9 58191997 IC50 = 39 nM T14597 CT3EW2 59292007 IC50 > 1000 nM T14597 CHC3W6 59484610 IC50 = 29 nM T14597 C1B3NR 59484612 IC50 = 100 nM T14597 CX0KC2 59484694 IC50 = 65 nM T14597 CXJ63M 59603829 IC50 > 100000 nM T14597 CQEU96 59603842 IC50 = 1000 nM T14597 C10AMI 66553589 IC50 > 10000 nM T14597 CWI6K5 67035106 IC50 > 10000 nM T14597 C38RGB 67035556 IC50 > 10000 nM T14597 CV63UL 67240318 IC50 > 10000 nM T14597 C8I7GC 68293638 IC50 > 10000 nM T14597 CD56XK 68293660 IC50 > 10000 nM T14597 C57ENP 68629464 IC50 = 0.92 nM T14597 CG7KR4 68669354 IC50 = 4.1 nM T14597 C5DGR9 69036886 IC50 = 10000 nM T14597 CWYG39 70684700 Ki = 3100 nM T14597 CYP97H 70688851 IC50 = 6500 nM T14597 CEQP73 70690935 IC50 = 4800 nM T14597 CUT1L7 70693079 IC50 > 10000 nM T14597 CQ5W6D 70693519 IC50 = 46 nM T14597 C6W1NL 71244639 IC50 = 1574 nM T14597 C5RE4T 71244643 IC50 = 324.4 nM T14597 CQ6A9L 71244644 IC50 = 1536 nM T14597 C1LH2U 71449341 IC50 = 8.5 nM T14597 C4BXY8 71449342 IC50 = 14 nM T14597 CEBO91 71452977 IC50 = 11 nM T14597 CJ2L8G 71455836 IC50 = 3000 nM T14597 CKT60L 71455860 Ki > 1400 nM T14597 CCGJ48 71456241 IC50 = 966 nM T14597 C7X4MD 71456750 IC50 > 25000 nM T14597 CTWX94 71457629 IC50 > 40000 nM T14597 C3AEL4 71457630 IC50 > 40000 nM T14597 C4V6TN 71459522 IC50 > 40000 nM T14597 CXMH59 71508796 IC50 = 2380 nM T14597 CJ0VS6 71508797 IC50 = 850 nM T14597 C6C4XN 71508798 IC50 = 180 nM T14597 C9F4SA 71508839 IC50 = 2230 nM T14597 COH1C9 71508888 IC50 = 1320 nM T14597 CMQ42Y 71508889 IC50 = 460 nM T14597 C9DIK2 71512060 IC50 = 75 nM T14597 CF05BU 71513157 IC50 = 149.4 nM T14597 CS1ZX0 71513822 IC50 = 1.38 nM T14597 CW6DN0 71514054 IC50 = 97.1 nM T14597 CXRK32 71519007 IC50 > 200 ug.mL-1 T14597 CI2Z5Y 71519008 IC50 = 96 ug.mL-1 T14597 CJ4KV6 71519009 IC50 > 200 ug.mL-1 T14597 C42MFK 71519172 IC50 = 40 ug.mL-1 T14597 C3XP1F 71519173 IC50 = 80 ug.mL-1 T14597 CC89QU 71519174 IC50 > 200 ug.mL-1 T14597 CGY2N8 71519175 IC50 > 200 ug.mL-1 T14597 C7RG1Z 71519338 IC50 = 46 ug.mL-1 T14597 COFB13 71519339 IC50 = 35 ug.mL-1 T14597 CJE5N6 71519340 IC50 = 63 ug.mL-1 T14597 CG0N8I 71519341 IC50 = 37 ug.mL-1 T14597 CM4PG6 71519493 IC50 > 200 ug.mL-1 T14597 CVUP53 71524867 IC50 = 7240 nM T14597 CQ52FW 71524868 IC50 = 10630 nM T14597 CQ7L5U 71524869 IC50 = 5460 nM T14597 CVPO31 71524870 IC50 = 9150 nM T14597 CSM8Q3 71524871 IC50 = 4180 nM T14597 CHZA07 71524872 IC50 = 6680 nM T14597 CW9M5E 71524873 IC50 = 6840 nM T14597 C75GEB 71524914 IC50 = 5690 nM T14597 CO1H9P 71524915 IC50 = 1750 nM T14597 CNZF95 71524916 IC50 = 3590 nM T14597 CXP7G2 71524917 IC50 = 3070 nM T14597 CQR8V0 71524918 IC50 = 2320 nM T14597 CQ34CK 71524919 IC50 = 3010 nM T14597 C12GMV 71524960 IC50 = 1980 nM T14597 C7BU0K 71524961 IC50 = 2010 nM T14597 C4R6CL 71524962 IC50 = 3870 nM T14597 CQ7UT5 71524963 IC50 = 1210 nM T14597 CRO0N8 71524964 IC50 = 3280 nM T14597 CZQ2S4 71524965 IC50 = 1040 nM T14597 C8A9IN 71525006 IC50 = 880 nM T14597 CH8LC0 71525007 IC50 = 1280 nM T14597 CT47DK 71525008 IC50 = 1450 nM T14597 C0M4LC 71525009 IC50 = 1020 nM T14597 C1SFD7 71532857 IC50 = 190 ug.mL-1 T14597 C8U9MB 71532907 IC50 = 27 ug.mL-1 T14597 COQ5V1 71532908 IC50 = 18 ug.mL-1 T14597 CE9N2D 71532909 IC50 = 22 ug.mL-1 T14597 CB3SO2 71567006 IC50 > 10000 nM T14597 CDJY72 71568837 IC50 > 10000 nM T14597 CRX81Q 71575642 IC50 > 10000 nM T14597 C1BCX0 71579696 IC50 > 1000 nM T14597 CZ31PU 71583657 IC50 = 24 nM T14597 C6RS7H 71583658 IC50 = 30 nM T14597 CWD2Z5 71585566 IC50 = 319 nM T14597 CQX8L3 71616700 IC50 = 180 nM T14597 CE6QA1 71616701 IC50 = 890 nM T14597 C4ZDO0 71616702 IC50 = 82 nM T14597 C03HCR 71616703 IC50 = 6000 nM T14597 CWTH52 71616704 IC50 = 1300 nM T14597 CZ7XB4 71616807 IC50 = 1100 nM T14597 CH2RA9 71658877 IC50 > 10000 nM T14597 CJI05L 71658878 IC50 > 10000 nM T14597 CCS41V 71658995 IC50 > 10000 nM T14597 CI91ZX 71658997 IC50 > 10000 nM T14597 CL9T2I 71658998 IC50 > 10000 nM T14597 C9Z0KG 71726907 IC50 = 8.5 nM T14597 CNY9K7 71765762 IC50 = 59 nM T14597 CEG6O2 72163258 IC50 = 360 nM T14597 CSM72B 72163259 IC50 = 860 nM T14597 C6VGD3 72163260 IC50 = 550 nM T14597 CE98SI 72163261 IC50 = 230 nM T14597 C0D8KH 72163262 IC50 = 250 nM T14597 CUO10A 72163263 IC50 = 1100 nM T14597 C4JM2F 72163401 IC50 = 1500 nM T14597 CUG3Z1 72165162 IC50 = 110 nM T14597 CIU90H 72202607 IC50 = 73 nM T14597 C60TUV 72737208 IC50 = 112 nM T14597 CJ3WA6 72737404 IC50 = 78 nM T14597 CP58UB 73053605 IC50 = 250 nM T14597 C9EXR4 73351100 IC50 = 8.6 nM T14597 CXC0O2 73352566 IC50 = 18.3 nM T14597 CZJ2S7 73352567 IC50 = 15.9 nM T14597 CCI47S 73352568 IC50 = 3.9 nM T14597 C83XBD 73354112 IC50 = 996 nM T14597 CF9A7B 74766095 IC50 = 55 nM T14597 CP5C7Y 76311266 IC50 = 1240 nM T14597 C4GD6X 76311267 IC50 = 390 nM T14597 C9XZ0C 76311268 IC50 = 29 nM T14597 C29NOJ 76314857 IC50 = 689 nM T14597 CQT97B 76314858 IC50 = 376 nM T14597 C27JRQ 76317764 IC50 = 290 nM T14597 C8AJ3M 76317765 IC50 = 230 nM T14597 CIV6B3 76318467 IC50 = 54800 nM T14597 C4PRL2 76318468 IC50 = 28300 nM T14597 CFTP19 76318469 IC50 = 576 nM T14597 CQ01AS 76318470 IC50 = 91200 nM T14597 CJE4B1 76321478 IC50 = 1110 nM T14597 CG67DB 76321482 IC50 = 930 nM T14597 CV0C8D 76322137 IC50 = 1150 nM T14597 C3QMZ9 76325759 IC50 = 978 nM T14597 C65WFX 76325760 IC50 = 66 nM T14597 CWG41I 76325761 IC50 = 6530 nM T14597 CV9H0X 76329340 IC50 = 1150 nM T14597 CJKG82 76329341 IC50 = 8830 nM T14597 CCP9B2 76329342 IC50 = 978 nM T14597 CX8Q2U 76329343 IC50 = 298 nM T14597 C0BJ8F 76332331 IC50 = 290 nM T14597 CY1N5G 76332981 IC50 = 13 nM T14597 CXBD37 76332982 IC50 = 1640 nM T14597 CJ2T9E 76332983 IC50 = 1300 nM T14597 CL0UZ2 76332984 IC50 = 310 nM T14597 C4J5BS 76335961 IC50 = 250 nM T14597 CG56FE 76335963 IC50 = 330 nM T14597 C4HOM3 76900440 IC50 = 1036 nM T14597 CNA52Z 78324176 IC50 = 674 nM T14597 C90PJT 78324177 IC50 = 384 nM T14597 CEDG87 78324478 IC50 = 337 nM T14597 CQA2Y0 78324481 IC50 = 250 nM T14597 CCJ43A 86302281 IC50 = 40 nM T14597 CB5NJ4 86302541 IC50 > 10000 nM T14597 CPG3A5 86302574 IC50 > 30000 nM T14597 C1HW4B 89735655 IC50 > 100000 nM T14597 CPH85G 90322858 IC50 = 344 nM T14597 CX29IY 90655145 IC50 = 30 nM T14597 CO7W1V 90662817 IC50 = 4500 nM T14597 CRL86F 90665697 IC50 > 1000 nM T14597 C9V6FU 90666397 IC50 > 1000 nM T14597 C5Q8VO 90666398 IC50 > 1000 nM T14597 CIB1E8 90666399 IC50 > 1000 nM T14597 C08ANK 90666400 IC50 > 1000 nM T14597 CL0KH2 90666401 IC50 > 1000 nM T14597 C9XI3E 90666402 IC50 > 1000 nM T14597 CLF29C 90666403 IC50 > 1000 nM T14597 CU9XB7 90666404 IC50 > 1000 nM T14597 CCL19D 90666405 IC50 > 1000 nM T14597 CYVM38 90666406 IC50 > 1000 nM T14597 CMY4T0 90666407 IC50 > 1000 nM T14597 CNE54X 90666408 IC50 > 1000 nM T14597 CF6Q9X 91669170 IC50 = 200 nM T14597 CWF97Y 92045039 IC50 = 16 nM T14597 CIU05O 118710979 IC50 = 14800 nM T14597 CJL49M 118710980 IC50 = 8900 nM T14597 C8WL4B 118710981 IC50 = 19300 nM T14597 C7WCP5 118710982 IC50 = 1900 nM T14597 C8PE2Y 118710983 IC50 = 5200 nM T14597 CBGV74 118710984 IC50 = 2100 nM T14597 CN38JS 118710985 IC50 = 9000 nM T14597 C51LZM 118710986 IC50 = 4100 nM T14597 CU3KJ9 118710987 IC50 = 800 nM T14597 C05DOU 118710988 IC50 = 22700 nM T14597 CW8JQ2 118712118 IC50 = 5200 nM T14597 C46QUT 118717614 IC50 = 58.6 nM T14597 CJC34Y 118717615 IC50 = 48.3 nM T14597 CFEP93 118717616 IC50 = 52.2 nM T14597 CEC4H0 118717617 IC50 = 152 nM T14597 CU2TG3 118717618 IC50 = 163.8 nM T14597 C5OL0W 118717619 IC50 = 158.2 nM T14597 C3KLI5 118723185 IC50 > 100000 nM T14597 C65JUN 118725950 IC50 = 12370 nM T14597 CDBZ85 118738351 IC50 = 13.1 nM T14597 CJV62R 118738352 IC50 = 23.7 nM T14597 CSTB45 118738353 IC50 = 12.3 nM T14597 CM38XC 118738354 IC50 = 14.4 nM T14597 C1EDA6 118738355 IC50 = 19.8 nM T14597 C63SVY 118738356 IC50 = 6.8 nM T14597 CQ83JA 118738357 IC50 = 53.3 nM T14597 CUY8Z3 118900244 IC50 = 131.6 nM T14597 CB85RT 118900245 IC50 = 83.84 nM T14597 CR2X9A 118900269 IC50 = 261.8 nM T14597 CH3I9B 118900282 IC50 = 39.26 nM T14597 CI3TK4 118900289 IC50 = 10.94 nM T14597 C7V3DH 118900298 IC50 = 42.11 nM T14597 C0LIS1 118900305 IC50 = 148.3 nM T14597 CINT13 118900306 IC50 = 482.1 nM T14597 C4X7SD 122192466 IC50 > 10000 nM T14597 CC5KB6 122195541 IC50 = 77 nM T14597 CKG14J 122195542 IC50 = 706 nM T14597 CIPZ05 122195677 IC50 = 26.8 nM T14597 C4V5WK 122195678 IC50 = 625 nM T14597 C03XJB 122195679 IC50 > 10000 nM T14597 C2CM8S 122195680 IC50 = 126 nM T14597 CIC6N1 122195681 IC50 = 1390 nM T14597 C3F1YP 122195682 IC50 = 1000 nM T14597 C4IMA2 122195683 IC50 > 10000 nM T14597 C8TK1W 122195684 IC50 = 5050 nM T14597 C4FXV5 122195685 IC50 = 3290 nM T14597 C47QYW 122195686 IC50 > 10000 nM T14597 CZC4K1 122195687 IC50 = 2720 nM T14597 CK0Q3A 122195688 IC50 = 8000 nM T14597 CLTG90 122195689 IC50 = 275 nM T14597 C0TX3A 122195690 IC50 = 855 nM T14597 C52BMS 122195691 IC50 > 10000 nM T14597 C8KXV1 127025843 IC50 > 1000 nM T14597 CKS28E 127034802 IC50 > 1000 nM T14597 CKX40V 127037812 IC50 > 10000 nM T14597 C70RUP 127038480 IC50 > 10000 nM T14597 CEG89U 127038628 IC50 = 18890 nM T14597 C18SAK 127039275 IC50 = 3450 nM T14597 C5GJ1F 127039276 IC50 = 8270 nM T14597 CYNR48 127039277 IC50 = 510 nM T14597 C87AFX 127039599 IC50 = 5620 nM T14597 CUVR09 127039608 IC50 = 17250 nM T14597 COE17A 127039609 IC50 = 12050 nM T14597 C93XHQ 127039610 IC50 = 14040 nM T14597 CXLQ81 127039662 IC50 = 17000 nM T14597 CKT2I9 127039915 IC50 = 18120 nM T14597 CEQA86 127039935 IC50 = 2060 nM T14597 CTK6W3 127039936 IC50 = 3530 nM T14597 CB3X9Y 127039944 IC50 = 14930 nM T14597 CAL3D1 127039945 IC50 = 4100 nM T14597 CB5KT1 127039946 IC50 = 9960 nM T14597 C8PK1U 127040288 IC50 = 4070 nM T14597 CT4U6D 127040940 IC50 = 8540 nM T14597 CJ8E7C 127040941 IC50 = 2750 nM T14597 CA6RH0 127040942 IC50 = 12660 nM T14597 CP6D1T 127040943 IC50 = 13160 nM T14597 C3WCN8 127041777 IC50 > 10000 nM T14597 CP15ZX 127043295 IC50 = 676 nM T14597 CV0F3N 127045112 IC50 = 1350 nM T14597 CTPY32 127045266 IC50 = 874 nM T14597 CWI8Q2 127045267 IC50 = 590 nM T14597 CV5I8S 127045270 IC50 = 1202 nM T14597 CHK16Q 127045929 IC50 > 1000 nM T14597 CY3J0C 127047591 IC50 > 1000 nM T14597 CDL7Z4 127048297 IC50 = 19.2 nM T14597 CPH4B3 127048979 IC50 = 32.3 nM T14597 CB3G8V 127050557 IC50 = 12.1 nM T14597 C9XM4K 127052093 IC50 = 33.1 nM T14597 C5N0QK 127052408 IC50 = 40.6 nM T14597 CIU72D 127264586 IC50 = 8.1 nM T14597 CUO0C5 132156633 IC50 > 10000 nM T14597 C0G9TV 132495274 IC50 = 174.9 nM T14597 CL6E4J 132601725 IC50 > 25000 nM T14597 CM5T6K 134130825 IC50 = 5 nM T14597 CC1EB5 134131929 IC50 = 27 nM T14597 CHW59N 134132187 IC50 = 77 nM T14597 CA7J2D 134132574 IC50 = 16.4 nM T14597 CS79UR 134133060 IC50 = 1100 nM T14597 CMZG34 134133313 IC50 = 102 nM T14597 C1VOY4 134133329 IC50 = 33 nM T14597 CX2WN6 134134364 IC50 = 38 nM T14597 CTZ84R 134134811 IC50 = 3200 nM T14597 CSZX25 134135323 IC50 = 53 nM T14597 CDMJ75 134135414 IC50 = 706.7 nM T14597 CUL3Q0 134136044 IC50 = 1300 nM T14597 C1GVQ7 134136098 IC50 = 556 nM T14597 C3G7TQ 134136245 IC50 = 30 nM T14597 CZD0J5 134136450 IC50 = 4700 nM T14597 CL4PT1 134137211 IC50 > 10000 nM T14597 CYGZ85 134137500 IC50 > 1000 nM T14597 CJC1E8 134137789 IC50 > 1000 nM T14597 CJ7C1N 134137974 IC50 = 14 nM T14597 C2L8OB 134138134 IC50 = 230 nM T14597 C3RA6C 134138227 IC50 = 386.1 nM T14597 CY3U6V 134138310 IC50 = 404 nM T14597 C4QSZ5 134138566 IC50 = 413 nM T14597 CZU97C 134138682 IC50 = 12 nM T14597 C6RGN8 134138812 IC50 = 100 nM T14597 C58FUC 134139047 IC50 = 406 nM T14597 CA7PD8 134139534 IC50 > 1000 nM T14597 C3OBC6 134139548 IC50 > 1000 nM T14597 CW69GT 134139694 IC50 = 23 nM T14597 CQE08L 134139702 IC50 = 89 nM T14597 CK7EZ2 134139706 IC50 > 1000 nM T14597 CO9W1Q 134139995 IC50 = 9 nM T14597 C8JR1X 134140108 IC50 = 19 nM T14597 CCF0X1 134140501 IC50 = 165.5 nM T14597 C6UJG4 134140680 IC50 = 815 nM T14597 CI2L7Z 134140949 IC50 = 958 nM T14597 CC3I0G 134142769 IC50 > 10000 nM T14597 CI92TY 134142809 IC50 = 6200 nM T14597 C4F6VU 134143525 IC50 = 128 nM T14597 C1OYR9 134145751 IC50 = 419 nM T14597 CRZ0E5 134146010 IC50 = 19 nM T14597 CZP47U 134146163 IC50 = 120 nM T14597 CN35SO 134146628 IC50 > 1000 nM T14597 CHJ13S 134146699 IC50 = 19 nM T14597 C0KNV3 134146887 IC50 = 62 nM T14597 C4U8KT 134147234 IC50 = 30 nM T14597 CJ1FQ6 134147869 IC50 = 62 nM T14597 CXS38A 134147887 IC50 = 32 nM T14597 CPGL96 134148137 IC50 = 153 nM T14597 CN4HT6 134148374 IC50 = 1600 nM T14597 C5R2PK 134148588 IC50 = 290 nM T14597 C0AWH3 134148660 IC50 = 20 nM T14597 CP14DK 134149339 IC50 = 537.4 nM T14597 CRBI31 134149577 IC50 = 180 nM T14597 C6Z2JL 134149963 IC50 = 782 nM T14597 CE69LC 134150331 IC50 = 11 nM T14597 CQ03OC 134150381 IC50 = 21 nM T14597 CJ56EZ 134150417 IC50 = 2 nM T14597 CM7H0R 134150543 IC50 = 192.8 nM T14597 CQK40B 134150618 IC50 = 17 nM T14597 CA4SQ5 134151152 IC50 = 800 nM T14597 C7CT2Y 134151327 IC50 = 642 nM T14597 CI4A1T 134152401 IC50 = 278 nM T14597 C0N6JF 134152887 IC50 = 100 nM T14597 C9ORY0 134152991 IC50 = 124 nM T14597 CLBK62 134153313 IC50 = 798 nM T14597 C6JFN5 134153988 IC50 = 198 nM T14597 CET5R1 134154580 IC50 > 10000 nM T14597 C5YX7T 134154596 IC50 = 19 nM T14597 C07RWN 134154721 IC50 = 174 nM T14597 CV5M1T 134154754 IC50 = 4 nM T14597 CI0S4B 134155078 IC50 = 458 nM T14597 CMH0X4 134155167 IC50 = 897 nM T14597 C48UIX 134155220 IC50 = 509 nM T14597 C9DRQ6 134155700 IC50 = 10 nM T14597 C90IBM 134155874 IC50 > 10000 nM T14597 C6HN5J 134155932 IC50 = 35 nM T14597 CBY2R8 134156011 IC50 = 176.7 nM T14597 CNG41Q 134156713 IC50 > 10000 nM T14597 CQD93J 134156816 IC50 = 45 nM T14597 C3HCT6 134156845 IC50 = 42 nM T14597 CI4W7T 134156856 IC50 > 1000 nM T14597 COVM37 134157236 IC50 = 3900 nM T14597 CEHV70 134157345 IC50 = 35 nM T14597 CG36DX 134157614 IC50 = 286 nM T14597 C7EMI6 135236457 IC50 = 730 nM T14597 CXDY80 135236566 IC50 = 167 nM T14597 CIOD87 135236597 IC50 = 590 nM T14597 CB6EG0 135236676 IC50 > 10000 nM T14597 C0DV1Q 135236809 IC50 = 730 nM T14597 CS4BM3 135236903 IC50 = 160 nM T14597 CGJ07D 135236905 IC50 = 93 nM T14597 CJ1I5M 135402981 IC50 > 1000 nM T14597 CH97JB 135402982 IC50 > 1000 nM T14597 C26GSU 135402983 IC50 > 1000 nM T14597 CK8EJ6 135402984 IC50 > 1000 nM T14597 CK9D4A 135428921 IC50 = 780 nM T14597 CIJ9Q2 135461535 IC50 = 6029 nM T14597 CV2RZ4 135464244 IC50 = 7.4 ug.mL-1 T14597 C3IJ9V 135497787 IC50 > 100000 nM T14597 C9YNE7 135497791 IC50 > 100000 nM T14597 C8HO5W 135497794 IC50 > 100000 nM T14597 CSP15M 135497800 IC50 > 100000 nM T14597 C0S3KJ 135497814 IC50 > 10000 nM T14597 CBF73U 135497834 IC50 = 3820 nM T14597 CEKY53 135497841 IC50 = 4170 nM T14597 C7GKS9 135497849 IC50 = 5120 nM T14597 C3WKV4 135497850 IC50 = 3600 nM T14597 CTUB09 135497851 IC50 = 140 nM T14597 COH6V1 135497852 IC50 = 1000 nM T14597 CU8T6K 135497853 IC50 = 240 nM T14597 CC58VR 135497854 IC50 = 85 nM T14597 C0ML5X 135497855 IC50 = 89 nM T14597 C1PJB2 135497865 IC50 > 100000 nM T14597 C1V9AZ 135497869 IC50 > 10000 nM T14597 CN2W4U 135497870 IC50 > 10000 nM T14597 C03EJP 135497876 IC50 = 6510 nM T14597 CR09SN 135497877 IC50 > 100000 nM T14597 CU6T8C 135497878 IC50 > 100000 nM T14597 C45KEI 135497879 IC50 > 100000 nM T14597 CK5G2W 135510524 IC50 = 1070 nM T14597 CTJ48K 135524085 IC50 = 9500 nM T14597 CUT1W7 135524168 IC50 > 10000 nM T14597 C2MAC7 135536640 IC50 > 100000 nM T14597 C19QOB 135620673 IC50 > 10000 nM T14597 C37RUJ 135620674 IC50 > 100000 nM T14597 CD08US 135620675 IC50 = 9300 nM T14597 CADG57 135620676 IC50 > 100000 nM T14597 C4XV9S 135620677 IC50 = 12000 nM T14597 CO9L3F 135620678 IC50 = 37000 nM T14597 C0IXJ4 135620680 IC50 > 100000 nM T14597 CZ49HM 135723775 IC50 = 3030 nM T14597 C6V4DX 135794286 IC50 > 10000 nM T14597 CO21NR 135823061 IC50 > 100000 nM T14597 CE95HA 135922389 IC50 = 32730 nM T14597 C3BZ4A 135922390 IC50 > 100000 nM T14597 C2PAV1 135971426 IC50 > 10000 nM T14597 CLN6Y8 136026516 IC50 > 100000 nM T14597 CFKB53 136104460 IC50 > 100000 nM T14597 C1Y0PS 136118031 IC50 > 100000 nM T14597 CA76XZ 136118032 IC50 > 100000 nM T14597 CVQ41X 136118033 IC50 > 100000 nM T14597 CU5XR2 136118034 IC50 > 100000 nM T14597 C4G6PT 136118035 IC50 > 100000 nM T14597 CGP69Y 136130281 IC50 = 1000 nM T14597 CDT7E4 136211077 IC50 > 1000 nM T14597 C3Z4AT 137321159 IC50 > 10000 nM T14597 CE75QD 137321162 IC50 > 10000 nM T14597 C25ERN 137631967 IC50 = 1 nM T14597 C8J5YE 137633149 IC50 > 100000 nM T14597 CWP23Z 137633367 IC50 = 8800 nM T14597 C2IOU5 137636607 IC50 = 3200 nM T14597 CT17QN 137636787 IC50 = 160 nM T14597 C06JRX 137637094 IC50 > 10 nM T14597 CE75PY 137639383 IC50 = 240 nM T14597 CHSF21 137642481 IC50 = 2400 nM T14597 CYIM43 137642492 IC50 = 52400 nM T14597 CS6J0V 137646549 IC50 = 910 nM T14597 C39ECO 137646754 IC50 = 45700 nM T14597 CB4G7L 137648004 IC50 = 2500 nM T14597 C3UBN8 137650330 IC50 = 4700 nM T14597 CR27SL 137650383 IC50 = 46800 nM T14597 CI1U0H 137650532 IC50 = 1200 nM T14597 CX12DJ 137650597 IC50 = 190 nM T14597 C1DK0P 137651391 IC50 = 1 nM T14597 C28QUP 137652864 IC50 = 1350 nM T14597 C9BF1E 137653143 IC50 = 36900 nM T14597 C6RWG4 137653308 IC50 = 6500 nM T14597 C5LV3R 137653430 IC50 = 2100 nM T14597 CBUK30 137656424 IC50 = 52600 nM T14597 COZA85 137656751 IC50 = 610 nM T14597 CV5H3Z 137657932 IC50 = 1 nM T14597 CW59EN 137658341 IC50 = 190 nM T14597 CR91LE 137659218 IC50 = 2700 nM T14597 C8NZ9V 137659669 IC50 = 1700 nM T14597 C98GQX 137660836 IC50 = 2500 nM T14597 CB72MA 137661754 IC50 = 57600 nM T14597 CSRI06 138547901 IC50 > 1000 nM T14597 CUXO19 138617501 IC50 > 1000 nM T14597 CCXG67 142735680 IC50 = 212 nM T14597 CO9P7G 145351804 IC50 > 1000 nM T14597 C6VB3O 145925651 IC50 >= 5000 nM T14597 C29XUO 145945978 IC50 > 1000 nM T14597 C3LW9D 145952066 IC50 = 10400 nM T14597 CKRP30 145952676 IC50 = 390 nM T14597 C6G4NF 145955071 IC50 = 9710 nM T14597 CLK9N3 145959197 IC50 = 25400 nM T14597 CHT30M 145959430 IC50 = 31500 nM T14597 CMC76F 145959984 IC50 = 18000 nM T14597 C9R0TU 145960317 IC50 = 760 nM T14597 C4OD9Q 145967187 IC50 = 23.2 nM T14597 CSJ0X9 145971962 IC50 = 300 nM T14597 CTA34O 145979089 IC50 = 240 nM T14597 CE31VG 145979714 IC50 > 10000 nM T14597 C9QFA1 145980052 IC50 = 1500 nM T14597 CLX91B 145981733 IC50 = 19200 nM T14597 CYUD47 145984188 IC50 = 100 nM T14597 CDM05I 145985073 IC50 = 100 nM T14597 C7A4WK 145988274 IC50 = 879 nM T14597 CDVL79 145988898 IC50 = 19 nM T14597 C9BX4U 145988956 IC50 > 10000 nM T14597 CWI75O 145990017 IC50 = 96 nM T14597 C2PBJ5 145990245 IC50 = 37100 nM T14597 COU0E6 145991881 IC50 = 1200 nM T14597 CE10PX 155512047 IC50 = 212 nM T14597 CL4B2M 155512535 IC50 = 64 nM T14597 C81YCJ 155513061 IC50 = 54 nM T14597 C2MD1Q 155513187 IC50 > 10000 nM T14597 C7SK0E 155513959 IC50 = 9.6 nM T14597 C86HPW 155518524 IC50 = 24000 nM T14597 C3NA2I 155519537 IC50 > 1000 nM T14597 C5EZR1 155524215 IC50 = 209 nM T14597 C8I3SW 155527677 IC50 = 225 nM T14597 CJ6T5H 155533092 IC50 = 78 nM T14597 C78MZC 155536330 IC50 = 37 nM T14597 CP8ZV6 155538283 IC50 = 67 nM T14597 CE46SL 155540854 IC50 = 2280 nM T14597 C5O4JM 155540856 IC50 = 6960 nM T14597 C02VLJ 155542715 IC50 = 54 nM T14597 CTQ9S4 155543012 IC50 = 2.1 nM T14597 CEDT28 155552106 IC50 = 471 nM T14597 CGVU70 155554426 IC50 > 30000 nM T14597 C2Q8OK 155559257 IC50 = 158 nM T14597 CC5F3I 155562216 IC50 = 104 nM T14597 CY1KP0 155564719 IC50 = 59 nM T14597 CBS5F3 155564756 IC50 = 90 nM T14597 CWAF51 155566440 IC50 = 448 nM T14597 D00ATA 5908088 IC50 > 100000 nM T14597 D00ERW 44444843 Ki > 1438 nM T14597 D00HVA 11624601 Ki > 1400 nM T14597 D00TJF 11807783 IC50 = 3290 nM T14597 D00TZD 2776 IC50 = 378 nM T14597 D00VZA 5328763 IC50 = 18000 nM T14597 D01NTW 5328768 IC50 = 6400 nM T14597 D01OKF 46207013 IC50 = 1880 nM T14597 D01RHR 71519693 IC50 = 19 nM T14597 D01VFR 4708 IC50 = 5.7 nM T14597 D01WYI 9995195 IC50 = 2.2 nM T14597 D02ARA 44279279 IC50 = 1300 nM T14597 D03ATU 4707 IC50 = 52000 nM T14597 D03OKV 9844320 IC50 > 1000 nM T14597 D05FFT 11566580 IC50 = 1.1 nM T14597 D05RFO 24180536 IC50 = 664 nM T14597 D06BJG 71556703 IC50 = 7 nM T14597 D06EHW 11625778 IC50 = 68 nM T14597 D06HVH 54613583 IC50 > 10000 nM T14597 D06QWO 14824655 IC50 > 10 ug.mL-1 T14597 D07OSK 6419834 IC50 > 100000 nM T14597 D08RZB 11153014 IC50 = 500 nM T14597 D09RFE 16216595 IC50 = 6600 nM T14597 D0A1CM 5281855 IC50 = 3540 nM T14597 D0A4XJ 5289418 IC50 > 100000 nM T14597 D0AY0F 70698427 IC50 > 10000 nM T14597 D0B7ZB 44437844 IC50 = 13500 nM T14597 D0B8DE 135469328 IC50 > 10000 nM T14597 D0C2SF 11183327 IC50 = 11000 nM T14597 D0D6MH 11617559 IC50 > 24000 nM T14597 D0EE6A 6398883 IC50 > 1000 nM T14597 D0G3SZ 6918469 IC50 > 10 ug.mL-1 T14597 D0H2DD 6411478 IC50 = 7900 nM T14597 D0HE0E 5941540 IC50 = 90200 nM T14597 D0HM5W 5328042 IC50 = 670 nM T14597 D0L0HG 766949 IC50 > 10000 nM T14597 D0M4SY 135440466 IC50 = 17100 nM T14597 D0NH7M 5328760 IC50 = 18000 nM T14597 D0P0IE 10205 IC50 = 30800 nM T14597 D0P0WT 3139 IC50 > 10000 nM T14597 D0Q3GG 667601 IC50 = 5700 nM T14597 D0Q3NG 11715520 Ki > 1400 nM T14597 D0S7IE 11658882 Ki > 1400 nM T14597 D0T9FQ 10061448 IC50 > 10000 nM T14597 D0UN9O 3385203 IC50 >= 10000 nM T14597 D0X4UE 10220590 IC50 = 6390 nM T14597 D0YZ7H 9797370 IC50 > 10000 nM T14597 D0Z4HV 10354294 IC50 > 10000 nM T14597 D0Z7TM 22273644 IC50 > 5000 nM T71374 D01ZRI 6450551 Ki = 4.2 nM T71374 D02XNW 5494449 Ki = 11 nM T71374 D0E3TC 44259 IC50 = 9.49 nM T71374 D0HB3F 118340554 IC50 = 3900 nM T71374 C63WLY 89644 IC50 = 2.5 ug.mL-1 T71374 C5JE2Z 104860 IC50 = 1.7 ug.mL-1 T71374 CI1NA5 159926 IC50 = 4.3 ug.mL-1 T71374 CYBA43 177458 IC50 = 4.4 ug.mL-1 T71374 CUO5Y3 1020400 IC50 = 13000 nM T71374 C3L7YE 2077962 IC50 = 860 nM T71374 CDQ3M7 5359485 IC50 = 0.96 ug.mL-1 T71374 C54BYP 5360741 IC50 = 2.5 ug.mL-1 T71374 C36GHS 5735633 IC50 = 13000 nM T71374 CT8U7I 5874584 IC50 = 230 nM T71374 C34FPE 6510285 IC50 = 6100 nM T71374 CKIP13 7769752 IC50 = 860 nM T71374 CBOP58 11293798 Ki > 10000 nM T71374 C26BZX 11362471 Ki > 10000 nM T71374 CWXB93 11397177 Ki > 10000 nM T71374 CL7X4Q 11530963 IC50 = 990 nM T71374 CDGF78 15282555 IC50 = 4100 nM T71374 CFPW41 16007116 Ki > 4300 nM T71374 CCPS81 24764502 IC50 > 35000 nM T71374 C4V9GH 24894117 IC50 = 10000 nM T71374 CJH19T 24894883 IC50 = 9200 nM T71374 CJ14YB 24894884 IC50 = 12000 nM T71374 CHVU39 24894885 IC50 = 46000 nM T71374 C57BHF 24894888 IC50 = 35000 nM T71374 CB5TP8 24894992 IC50 = 28000 nM T71374 C38TGD 24894994 IC50 = 23000 nM T71374 CP7QT2 24894995 IC50 = 7700 nM T71374 C41SIT 24894996 IC50 = 44000 nM T71374 CFW40U 24894997 IC50 = 9000 nM T71374 CF4N9X 24895100 IC50 = 16000 nM T71374 CN13JF 24899915 IC50 = 0.38 ug.mL-1 T71374 CBWR97 24899916 IC50 = 0.83 ug.mL-1 T71374 C9F2JD 24899917 IC50 > 10 ug.mL-1 T71374 C64MTI 24900160 IC50 = 1.7 ug.mL-1 T71374 CO2I6Q 24900161 IC50 = 2.5 ug.mL-1 T71374 CJ5U1X 42639664 IC50 = 1.4 ug.mL-1 T71374 CS2VZ5 44230280 Ki = 100 nM T71374 CYH6P3 44520205 IC50 < 3 nM T71374 C3VRO9 44557921 IC50 > 10000 nM T71374 CY3HW5 46224684 IC50 = 380 nM T71374 CLS29B 46872626 IC50 > 10000 nM T71374 CU7SM4 53529356 IC50 = 6100 nM T71374 CD3SZ1 56959836 IC50 = 1.5 nM T71374 CF2QP6 56959838 IC50 = 20 nM T71374 CN2GI7 56959991 IC50 = 0.39 nM T71374 CB3I0R 56960132 IC50 = 0.64 nM T71374 CJO0V9 56960133 IC50 = 5.2 nM T71374 CT0U1H 58486131 IC50 = 4.6 nM T71374 CAW51G 58486138 IC50 = 0.9 nM T71374 C4Y6PF 58486151 IC50 = 5.9 nM T71374 CCF5Y4 58486156 IC50 = 1.5 nM T71374 C2I3QW 58486157 IC50 = 0.69 nM T71374 COTW45 58486166 IC50 = 1.7 nM T71374 C7ZKF5 58486186 IC50 = 0.94 nM T71374 CBF7L4 58486208 IC50 = 1.2 nM T71374 CM91GS 58486210 IC50 = 1.2 nM T71374 CQPU86 58486223 IC50 = 1.6 nM T71374 CB0Z6T 58486228 IC50 = 54 nM T71374 C3ZKB1 58486287 IC50 = 1.7 nM T71374 CRB42N 58486297 IC50 = 1.3 nM T71374 C51FBH 58486335 IC50 = 30 nM T71374 C35FWX 58486367 IC50 = 1000 nM T71374 CPF24Q 58486383 IC50 = 1.1 nM T71374 C6R4HK 58486387 IC50 > 50000 nM T71374 C2BGP3 59442302 Ki = 25 nM T71374 CV63UL 67240318 IC50 > 10000 nM T71374 C6D3QJ 67448476 IC50 = 0.45 nM T71374 C65XEF 67955686 IC50 = 2.1 nM T71374 C32TVX 68230798 IC50 = 130 nM T71374 CKT60L 71455860 Ki = 7 nM T71374 C47JPV 75202872 IC50 > 50000 nM T71374 CR70LI 90395752 IC50 = 3900 nM T71374 CGB54P 101902999 IC50 = 89 nM T71374 CG62HP 101903000 IC50 = 83 nM T71374 C3KLI5 118723185 IC50 > 100000 nM T71374 CLU74Q 118731287 IC50 = 1.5 nM T71374 CO8Z2N 129900111 IC50 = 82 nM T71374 CIP61L 134153498 IC50 = 43.5 nM T71374 CLSE63 135398512 Ki = 11 nM T71374 C0CM9H 135879715 IC50 = 2200 nM T71374 C01HMT 135932346 IC50 = 2.4 nM T71374 CYXR26 135985503 IC50 = 13 nM T71374 C4RL7Q 135985508 IC50 = 7.3 nM T71374 C8WIM5 135985510 IC50 = 0.32 nM T71374 C3M7EP 135985511 Ki = 22 nM T71374 CMQ5W9 135985512 IC50 = 2 nM T71374 CGM2H4 135988906 IC50 = 1.4 nM T71374 CA46HS 135988914 IC50 = 64 nM T71374 CSO48W 135988918 IC50 = 10000 nM T71374 CXM18S 135988925 IC50 = 54 nM T71374 C1ZT4N 135988927 IC50 = 1.4 nM T71374 CJE79B 135988932 IC50 = 220 nM T71374 CODL21 135988938 IC50 = 540 nM T71374 CVG5B9 135988940 IC50 = 60 nM T71374 C68JXP 135988944 IC50 = 0.82 nM T71374 CG23XF 135988947 IC50 = 0.9 nM T71374 CIFX04 135988950 IC50 = 0.45 nM T71374 CGP53C 135988956 IC50 = 1300 nM T71374 CLNJ17 135988957 IC50 = 13 nM T71374 C7NU6A 135988961 IC50 = 2.3 nM T71374 CR81AC 135988980 IC50 = 0.48 nM T71374 C86BZJ 135988997 IC50 = 2 nM T71374 C80PXZ 135989011 IC50 = 1200 nM T71374 CC6SO7 135989013 IC50 = 42 nM T71374 C5BDV8 135989018 IC50 = 490 nM T71374 CD7L3X 135989019 IC50 = 29 nM T71374 CZ7EX0 136183413 IC50 = 3820 nM T71374 CY57SZ 136239319 IC50 = 47 nM T71374 CJ2L3P 136239450 IC50 = 390 nM T71374 C7XY0Q 136239451 IC50 = 240 nM T71374 CN5LQ2 136239452 IC50 = 6300 nM T71374 CY08AS 136244133 IC50 = 1.6 nM T71374 CFQO70 136375226 IC50 = 2.4 nM T71374 CC8Q2D 136375233 IC50 = 230 nM T71374 D06QWO 14824655 IC50 > 10 ug.mL-1 T71374 D08JPU 3501 Ki = 3.4 nM T71374 D0A1CM 5281855 IC50 = 2970 nM T71374 D0G3SZ 6918469 IC50 = 3.2 ug.mL-1 T71374 D0Z5TQ 5924208 IC50 = 230 nM T89736 D04AIT 5280445 IC50 = 20000 nM T89736 D07EXH 359 IC50 > 200000 nM T89736 D07MGA 72281 IC50 = 8300 nM T89736 D0J9ZR 4477 IC50 = 40000 nM T89736 D0K8KX 5280343 IC50 = 8100 nM T89736 C5H9TY 14697 IC50 = 207000 nM T89736 C3I7VB 102678 IC50 = 24500 nM T89736 CL5Y4J 159516 Ki = 3100 nM T89736 CV0B7W 442027 IC50 = 49600 nM T89736 C1E2FR 442048 IC50 = 283500 nM T89736 CZ3MD8 647122 IC50 = 16100 nM T89736 C2C8QU 948801 Ki = 27500 nM T89736 CXA4P6 1265413 IC50 = 90720 nM T89736 CUD4A1 1328543 IC50 = 58350 nM T89736 C3ZP4U 2131972 Ki = 9110 nM T89736 CA1N3H 2131982 Ki = 9930 nM T89736 CKL8B2 2219105 IC50 = 29900 nM T89736 CN43XQ 2806068 IC50 = 160 nM T89736 C5J6MO 2849659 IC50 = 28800 nM T89736 CN3P7A 2911959 IC50 = 74500 nM T89736 CZDG23 2947583 IC50 = 186000 nM T89736 CBIP72 2986413 IC50 = 76700 nM T89736 CCU3P7 3635406 IC50 = 2200 nM T89736 CZF0R5 4004950 IC50 = 500 nM T89736 C3AN7C 4117477 IC50 = 1180 nM T89736 CS2WB7 4236803 IC50 = 29800 nM T89736 C0AW3N 4378077 IC50 = 13860 nM T89736 CO3Y0T 4614896 IC50 = 9910 nM T89736 CY68ZT 4788586 IC50 = 940 nM T89736 CTR4Q1 5320532 IC50 = 13300 nM T89736 CVG47I 5958938 IC50 = 10500 nM T89736 CD8ZT2 6026688 IC50 > 50000 nM T89736 C3LZX9 8027611 IC50 = 12660 nM T89736 CJ4C5K 9180583 IC50 = 10800 nM T89736 CYQ8Z4 9882716 IC50 > 50000 nM T89736 C8K2NO 10062715 IC50 = 800000 nM T89736 C49CMU 10411574 IC50 = 21700 nM T89736 C6GN2F 11642725 IC50 = 870000 nM T89736 CHYP53 12310492 IC50 = 233400 nM T89736 C65EOH 15949840 IC50 = 7500 nM T89736 C9V8EM 15956553 IC50 = 300000 nM T89736 C3WYR4 16061499 IC50 = 2000 nM T89736 CTO43V 16085283 Ki = 116000 nM T89736 CU35DQ 21582568 IC50 = 220800 nM T89736 CN45FL 23427055 IC50 = 164700 nM T89736 CK3AF8 25256829 IC50 = 5400 nM T89736 C2SZ7L 42624533 IC50 = 14000 nM T89736 CYP8V1 44404067 IC50 > 50000 nM T89736 CD20PF 44433696 IC50 = 80000 nM T89736 CI4P2V 44433697 IC50 = 10000 nM T89736 CW7B0J 44433698 IC50 = 15000 nM T89736 C8DWL3 44433699 IC50 = 200000 nM T89736 C0ZPE2 44517748 IC50 = 2700 nM T89736 C0OH2T 44584893 IC50 = 5400 nM T89736 C0NZ5E 44584944 IC50 = 7300 nM T89736 CT70DZ 44590821 IC50 = 22500 nM T89736 C0SW2K 45266425 IC50 = 2500 nM T89736 C5WBP2 45266482 IC50 = 3800 nM T89736 CA4K8F 45266488 IC50 = 6600 nM T89736 C3BHZ4 45268445 IC50 > 50000 nM T89736 CC05NI 45268452 IC50 = 15400 nM T89736 C6QD9E 45269292 IC50 > 50000 nM T89736 CY7RV4 45269761 Ki = 21000 nM T89736 CO80TH 45269762 Ki = 297000 nM T89736 CU34ZK 45269763 Ki = 584000 nM T89736 C9P3LZ 45269764 Ki = 478000 nM T89736 CXS19V 45269765 Ki = 45200 nM T89736 C3DY4T 45270971 IC50 > 50000 nM T89736 CR4WA8 45270979 IC50 = 20900 nM T89736 CM78GO 45271412 Ki = 462000 nM T89736 CC90BU 45271826 IC50 = 5200 nM T89736 C0B6KX 45271831 IC50 = 9300 nM T89736 CN85IQ 45271832 IC50 = 8100 nM T89736 C7IF2O 45272299 Ki = 363000 nM T89736 CZRV73 45272304 Ki = 34100 nM T89736 CGV14L 45272305 Ki = 112000 nM T89736 CVTL97 45272306 Ki = 2200 nM T89736 CAM89I 45273174 Ki = 135000 nM T89736 CZT67B 45273179 Ki = 614000 nM T89736 CHF4M5 45273180 Ki = 49300 nM T89736 CND1R3 45273184 Ki = 159000 nM T89736 C0V5WT 45273625 IC50 > 50000 nM T89736 C6OE7V 46784066 IC50 = 28300 nM T89736 C6LH5I 46881919 Ki = 800 nM T89736 CI2FO1 49870840 IC50 = 5500 nM T89736 CF2D0I 49870841 IC50 = 8400 nM T89736 CM52SZ 49870842 IC50 = 6800 nM T89736 C8Q2CZ 50885062 IC50 > 50000 nM T89736 CJ6KV7 52941131 IC50 = 13900 nM T89736 C8M2QD 52943127 IC50 = 24300 nM T89736 CQ84MD 52945913 IC50 = 12000 nM T89736 CJ1LG2 52945915 IC50 = 42000 nM T89736 CZ35DX 52945977 IC50 = 128900 nM T89736 CAB1Y3 52946772 IC50 = 163200 nM T89736 CO4R1B 52947200 IC50 = 18000 nM T89736 CC4X1O 52948928 IC50 = 137700 nM T89736 CMG4U7 52949213 IC50 = 10800 nM T89736 C0X5BL 58589722 IC50 = 76740 nM T89736 CY3CL6 71544384 IC50 = 610 nM T89736 CV3P2U 71544385 IC50 = 230 nM T89736 CJS60O 71571220 IC50 = 49000 nM T89736 C1AY0M 71571221 IC50 = 49000 nM T89736 CY21XB 71571222 IC50 = 4600 nM T89736 C1DX9H 71571223 IC50 = 39000 nM T89736 CKE2C3 73056463 IC50 > 100000 nM T89736 C9S8ZH 73056464 IC50 > 100000 nM T89736 CK9OI0 73056465 IC50 = 31710 nM T89736 C4D8LK 73056466 IC50 = 32080 nM T89736 CRY86G 73056467 IC50 = 34910 nM T89736 C3VS4F 73056760 IC50 = 10070 nM T89736 CYH1F4 73056761 IC50 = 51330 nM T89736 C2CRZ8 73056762 IC50 = 2250 nM T89736 CD4YR3 73056763 IC50 = 11830 nM T89736 C3P2OZ 73056764 IC50 = 67200 nM T89736 C1H8PX 73056765 IC50 = 82910 nM T89736 C8JO7B 73056766 IC50 = 13860 nM T89736 CCYE63 73057087 IC50 = 5520 nM T89736 C54JWM 73057088 IC50 = 39870 nM T89736 C8RBU6 73057089 IC50 = 1040 nM T89736 CEBH65 73057090 IC50 = 1690 nM T89736 C8M2DX 73057091 IC50 = 17820 nM T89736 CQ42AZ 73057092 IC50 = 2820 nM T89736 CPLJ64 73057388 IC50 = 4700 nM T89736 CIN5V0 76320984 IC50 = 4300 nM T89736 C05AYV 102341658 IC50 = 16400 nM T89736 C8S3CR 102341659 IC50 = 37500 nM T89736 C2G9CP 127043455 IC50 = 20200 nM T89736 CVZ4I3 127043641 IC50 = 6000 nM T89736 C7BST4 127043642 IC50 = 5800 nM T89736 CGO01F 127043643 IC50 > 50000 nM T89736 C2TU5A 127043644 IC50 = 6400 nM T89736 C0Y9IT 127043645 IC50 = 41200 nM T89736 CF3B1Z 127045220 IC50 = 11700 nM T89736 CIXJ94 127045221 IC50 = 8600 nM T89736 CQ1CT5 127045222 IC50 = 18700 nM T89736 CKRX04 127045227 IC50 = 30700 nM T89736 CDZ2E1 127045228 IC50 > 50000 nM T89736 CG3E9B 127045229 IC50 = 6700 nM T89736 CG6VR3 127045386 IC50 = 15700 nM T89736 CK9JE3 127045387 IC50 > 50000 nM T89736 CY1E4Z 127045392 IC50 > 50000 nM T89736 CK5PA4 127045393 IC50 = 44700 nM T89736 C34TWD 127045394 IC50 > 50000 nM T89736 C97MQC 127048409 IC50 = 20000 nM T89736 C41VRM 127048410 IC50 = 7500 nM T89736 CZ0B1R 127052510 IC50 = 10000 nM T89736 CRW05E 127052511 IC50 > 50000 nM T89736 CC3TX0 127052512 Ki = 72000 nM T89736 CIQ1U9 127052513 Ki = 41000 nM T89736 CI13JZ 135452883 IC50 = 10000 nM T89736 CG1KW5 135470831 IC50 = 77090 nM T89736 CH4Q6A 145964401 IC50 = 5500 nM T89736 CHU61S 145964420 IC50 = 42100 nM T89736 C6YCA8 145964710 IC50 = 28800 nM T89736 CV6F7L 145966788 IC50 = 2100 nM T89736 CBWX17 145967285 IC50 = 4300 nM T89736 COR9X3 145972736 IC50 = 3900 nM T89736 CQ0M2X 145972809 IC50 = 4100 nM T89736 CF95RZ 145972878 IC50 = 3200 nM T89736 CXI0D1 145975081 IC50 = 6300 nM T89736 CG84ZR 145975487 IC50 = 5100 nM T89736 C91FOT 145976006 IC50 = 5200 nM T89736 C3F4UH 145978039 IC50 = 8800 nM T89736 CL7FB0 2919450 IC50 = 62790 nM T89736 D00RIX 5280443 IC50 = 280800 nM T89736 D01XMM 4117383 IC50 = 4450 nM T89736 D08MZY 145937 Ki = 8200 nM T89736 D08UYP 3008868 Ki = 2400 nM T89736 D09BUG 10207 IC50 = 132000 nM T89736 D0L7AT 10480940 Ki = 19300 nM T89736 D0S0BN 130976 Ki = 10600 nM T89736 D0SY2M 5281708 IC50 = 105000 nM T89736 D0UQ6U 10569 IC50 = 189100 nM T89736 D0WA9S 10429214 IC50 = 146500 nM T37371 D0E3TC 44259 IC50 = 15.8 nM T37371 D03BNU 59604787 IC50 > 10000 nM T37371 D0T3ME 156422 IC50 > 30000 nM T37371 CACS26 11561968 Ki > 2000 nM T37371 CU0E8O 11690457 Ki > 1000 nM T37371 C7YG1N 24759534 IC50 = 37000 nM T37371 C8NA4L 53384644 IC50 > 30000 nM T37371 CXJ63M 59603829 IC50 > 100000 nM T37371 CQEU96 59603842 IC50 = 1500 nM T37371 C1MR8Q 60097495 IC50 > 1000 nM T37371 CV63UL 67240318 IC50 > 10000 nM T37371 C5DGR9 69036886 IC50 = 10000 nM T37371 C1HW4B 89735655 IC50 = 1400 nM T37371 CHJ70O 118960212 IC50 = 260 nM T37371 C2MD1Q 155513187 IC50 > 10000 nM T62151 D03SKR 2803 Ki > 100 nM T62151 D06OFS 68712 Ki < 10000 nM T62151 D0E1WI 3345 Ki = 5462 nM T62151 D0L4FS 5280961 IC50 = 900 nM T62151 CY58BM 1880 IC50 = 17000 nM T62151 CU86VK 54459 Ki < 10 nM T62151 C39DLT 70287 Ki = 50000 nM T62151 CMH58G 152923 Ki = 51000 nM T62151 CUA2H0 3084422 Ki = 33.11 nM T62151 C6IPM8 3391493 IC50 = 40000 nM T62151 CP7G8W 3596579 IC50 = 150 nM T62151 CW63PI 4118326 IC50 = 7000 nM T62151 C5K7QS 4198873 IC50 = 300 nM T62151 C5J1DA 4393018 Ki = 199.53 nM T62151 C5LGJ1 5282362 IC50 = 4500 nM T62151 CA51BY 9794143 Ki < 10000 nM T62151 C13MBI 9794144 Ki < 10000 nM T62151 CNZ7M2 9794264 IC50 = 41.7 nM T62151 C8MD5K 9797371 IC50 > 9000 nM T62151 C2PLU8 9819934 IC50 >> 9000 nM T62151 C43XWS 9843294 IC50 = 4000 nM T62151 CP25HN 9867778 IC50 = 13000 nM T62151 CUX4A2 9885593 IC50 = 3000 nM T62151 CGK1S3 9888593 IC50 = 10000 nM T62151 C8CWV9 9907990 IC50 = 2100 nM T62151 C85ICB 9998250 IC50 = 5000 nM T62151 CUIL41 10012705 Ki = 933.25 nM T62151 CL53TD 10176639 Ki < 10000 nM T62151 C39IDW 10193224 IC50 >> 9000 nM T62151 CDOU49 10219780 Ki < 10000 nM T62151 CL4R3I 10313366 Ki < 10000 nM T62151 C6W5DM 10333157 Ki = 7244.36 nM T62151 CS3XT5 10363696 Ki = 409 nM T62151 CUJ32V 10419932 Ki = 123.03 nM T62151 CC51PD 10432095 IC50 = 2000 nM T62151 C5DY8H 10442436 Ki = 6.026 nM T62151 CXFE98 10588013 Ki < 10000 nM T62151 CD7N1Y 10613705 IC50 = 450 nM T62151 CF4Y1O 10657832 Ki < 10000 nM T62151 CP2YR9 10687704 IC50 = 1700 nM T62151 C12CSD 10862798 IC50 >> 9000 nM T62151 CQ5H8V 10869223 Ki = 181.97 nM T62151 CG1P0O 10925737 IC50 = 5000 nM T62151 C6RME5 10926283 IC50 > 9000 nM T62151 CS2H7X 10949302 IC50 = 6500 nM T62151 CA8Q9Z 10987033 Ki = 144.54 nM T62151 C3VR2W 10997791 Ki = 100 nM T62151 CKV9C4 11002709 IC50 >> 9000 nM T62151 C8ZF6V 11011399 Ki = 7585.78 nM T62151 CA7IB5 11043720 Ki = 48977.88 nM T62151 CJ1QY8 11063180 Ki = 2511.89 nM T62151 CMV68C 11090565 IC50 > 9000 nM T62151 C1UGL3 11097489 Ki = 269.15 nM T62151 CRT6N5 11137887 Ki = 12589.25 nM T62151 C6SXJ0 11140033 Ki = 12589.25 nM T62151 CUQ1L4 11728663 IC50 > 9000 nM T62151 C7Z1VD 11732018 IC50 = 5300 nM T62151 CBGA07 11748522 IC50 = 1500 nM T62151 C4E0QO 11761097 IC50 >> 9000 nM T62151 CR1NT6 12632113 Ki = 123.03 nM T62151 CZ63DE 44269122 Ki = 2691.53 nM T62151 C89FEL 44269124 Ki = 302 nM T62151 CS3B6M 44309180 Ki = 22.91 nM T62151 CG6XI0 44340754 IC50 = 7000 nM T62151 CZ2X3A 44352155 Ki = 812.83 nM T62151 C67ZNM 44352207 Ki = 1621.81 nM T62151 CWFQ58 44363688 Ki = 437 nM T62151 CST17U 44363907 Ki = 1920 nM T62151 CZTA92 44363923 Ki = 126 nM T62151 CHGO26 44363938 Ki = 6.5 nM T62151 C5T9YE 135436602 IC50 = 20000 nM T62151 C2WA9R 135457295 IC50 = 30000 nM T62151 CHNA50 135471217 IC50 = 10000 nM T62151 CJR38B 135483618 IC50 = 9500 nM T62151 CKG25Y 135495099 IC50 = 3600 nM T62151 CT3M5A 135497038 IC50 = 12000 nM T62151 CCDS87 135499808 IC50 = 50000 nM T62151 C6VS7P 135514579 IC50 = 200 nM T62151 CR05TL 135516788 IC50 = 40000 nM T62151 CD2X0Y 135524872 IC50 = 9500 nM T62151 CX95EP 136092233 IC50 = 10000 nM T62151 D01KKU 5281894 IC50 = 120 nM T62151 D01UYI 5281607 IC50 = 1600 nM T62151 D05ZPO 1890 IC50 = 13000 nM T62151 D09BIV 6455104 Ki = 1.905 nM T62151 D0N9FH 10442227 Ki = 0.8913 nM T62151 D0O9UY 10469827 IC50 = 200 nM T62151 D0OC4B 5357479 IC50 = 500 nM T62151 D0S9YX 5280373 IC50 = 400 nM T62151 D0SY2M 5281708 IC50 = 14000 nM T62151 D0SY6C 5282073 IC50 = 30 nM T62151 D0Z7NC 33273 Ki = 2.512 nM T07403 D01TJY 53340771 IC50 > 10 nM T07403 D0Q5LF 9961766 IC50 = 433 nM T07403 D02WII 9912743 IC50 = 0.75 nM T07403 C8AQP3 741467 IC50 = 1000 nM T07403 CT1Z2Y 823530 IC50 = 2200 nM T07403 C28NSK 1817642 IC50 = 4100 nM T07403 C4U0BM 1878893 IC50 = 1300 nM T07403 C5JSA4 9801270 IC50 = 55.9 nM T07403 CY2NE9 9803540 IC50 = 734 nM T07403 CTZW25 9806910 IC50 = 42 nM T07403 CI51MD 9807891 IC50 > 100000 nM T07403 CK6A0I 9808598 IC50 = 6140 nM T07403 CCJ07G 9822539 IC50 = 39.6 nM T07403 C4KMF1 9824454 IC50 = 1320 nM T07403 C13KPA 9848051 Ki < 10000 nM T07403 C04PAT 9849697 IC50 > 100000 nM T07403 C2XD7P 9851886 IC50 = 8000 nM T07403 CN1R0K 9852055 IC50 > 100000 nM T07403 C53EJZ 9868509 IC50 = 72.2 nM T07403 C2ZAK6 9870468 IC50 = 190 nM T07403 CA03MS 9912398 IC50 = 170 nM T07403 CUH19P 9951966 IC50 = 45.3 nM T07403 C8AJ2G 9985610 IC50 = 102 nM T07403 C91KYI 9985909 IC50 = 10.6 nM T07403 C56RJO 10001383 IC50 = 7000 nM T07403 C9X4ME 10003581 IC50 = 9.9 nM T07403 C09DEP 10045632 IC50 = 6000 nM T07403 C8TE7O 10052250 IC50 = 376.9 nM T07403 CALU36 10075519 IC50 = 4.3 nM T07403 C71AIN 10077862 IC50 = 10700 nM T07403 C2UY1Z 10099823 IC50 = 1.92 nM T07403 C9GY3Z 10100204 IC50 = 27 nM T07403 CG9MW5 10100699 IC50 = 179 nM T07403 C3YZ2N 10116180 IC50 = 324 nM T07403 CHWL67 10118022 IC50 = 168 nM T07403 CL2Z0P 10118913 IC50 = 622 nM T07403 C8WS2G 10119516 IC50 = 5790 nM T07403 CG9U5C 10120896 IC50 = 849 nM T07403 CQ1YJ7 10138062 IC50 = 363 nM T07403 CVPQ90 10139365 IC50 = 179 nM T07403 CLG5S1 10141712 IC50 = 565 nM T07403 CT4NY2 10187032 IC50 = 1998 nM T07403 CE5V8W 10187715 IC50 = 97 nM T07403 CS2JU4 10188054 IC50 = 466 nM T07403 CVGM95 10188056 IC50 = 436 nM T07403 CQ7R9N 10188398 IC50 = 9220 nM T07403 CV01DN 10188683 IC50 = 257 nM T07403 CSJH35 10206665 IC50 = 21 nM T07403 CRH9F6 10210770 IC50 = 1260 nM T07403 CLZW43 10211418 IC50 = 94 nM T07403 C2FGD4 10229869 IC50 = 1900 nM T07403 CS69QU 10231058 IC50 = 168 nM T07403 CHB7A6 10231860 IC50 = 9180 nM T07403 C1FH9Q 10232974 IC50 = 96 nM T07403 CC28TW 10249554 IC50 = 7000 nM T07403 C5GEL4 10273950 IC50 = 687 nM T07403 C7KA3Y 10280825 IC50 = 1230 nM T07403 CTD53A 10281032 IC50 = 46 nM T07403 C2YKU9 10282280 IC50 = 22 nM T07403 C25TMF 10282625 IC50 = 536 nM T07403 CC92ST 10299878 IC50 = 820 nM T07403 CV75FS 10300040 IC50 = 220 nM T07403 C7B2QP 10300477 IC50 = 164 nM T07403 C1XO6Q 10301396 IC50 = 2.83 nM T07403 CMDY64 10304716 IC50 = 83 nM T07403 C1G6WY 10366133 IC50 = 110 nM T07403 C9FV3S 10371492 IC50 = 14 nM T07403 C6I8LC 10385477 IC50 = 9000 nM T07403 CT0KX3 10387865 IC50 = 50 nM T07403 COG4R0 10394110 IC50 = 2.98 nM T07403 C0IWH4 10413082 IC50 = 3546 nM T07403 CF83CY 10431881 IC50 = 7.09 nM T07403 CPO4V0 10458994 IC50 = 52.2 nM T07403 CQR6B8 10460375 IC50 = 646 nM T07403 C3PD9F 10481891 IC50 = 19 nM T07403 CQ3PB2 10545196 IC50 = 122000 nM T07403 CN8M6I 10604155 IC50 = 10 nM T07403 CWP63R 10710179 IC50 = 100000 nM T07403 CJQK52 11166204 IC50 = 250 nM T07403 CF0Q5M 11168346 IC50 = 4 nM T07403 CWE7R5 11168754 IC50 = 330 nM T07403 CY12UD 11177161 IC50 = 94 nM T07403 C3VA9H 11204176 IC50 = 2 nM T07403 C72DKJ 11212745 IC50 = 63 nM T07403 CN17WU 11213435 IC50 = 350 nM T07403 CAX6N8 11224267 IC50 = 110 nM T07403 CJU14K 11249992 IC50 = 3 nM T07403 CU6JK8 11258559 IC50 = 17 nM T07403 CMJD76 11271230 IC50 = 92 nM T07403 CGC54M 11272114 IC50 = 2 nM T07403 CT08ZV 11272553 IC50 = 3 nM T07403 C0GUA3 11296107 IC50 = 2 nM T07403 CA6EM9 11306407 IC50 = 610 nM T07403 CZRP50 11337796 IC50 = 1500 nM T07403 COF9P4 11340507 IC50 = 3 nM T07403 CW09GY 11341120 IC50 = 2 nM T07403 CAV42L 11364489 IC50 = 7 nM T07403 C4R3UP 11376484 IC50 = 5 nM T07403 CQ3K4D 11385630 IC50 = 19 nM T07403 C6BK8D 11387592 IC50 = 3 nM T07403 CY5B3Z 11408255 IC50 = 1400 nM T07403 C3MC5H 11441045 IC50 = 810 nM T07403 C0C9IQ 11442204 IC50 = 360 nM T07403 CW5CP6 11451270 IC50 = 710 nM T07403 CXIM19 11454676 IC50 = 230 nM T07403 CC9Q5T 11478436 IC50 = 1000 nM T07403 CE43BF 11487182 IC50 = 29 nM T07403 C78OKP 11495823 IC50 = 570 nM T07403 C3U7CQ 11512183 IC50 = 18 nM T07403 CAH69M 11547136 IC50 = 41 nM T07403 C91BTP 11555311 IC50 = 8 nM T07403 CLOP01 11555715 IC50 = 11 nM T07403 CL1PB2 11568832 IC50 = 13 nM T07403 CR6GM5 11569874 IC50 = 42 nM T07403 C5SO0J 11577165 IC50 = 16 nM T07403 CX9YO2 11678416 IC50 = 100 nM T07403 CQ5IV6 11752188 IC50 = 2 nM T07403 CT4D1K 11799915 IC50 = 59000 nM T07403 CFP4T1 12968380 IC50 = 54000 nM T07403 C5K9XD 12968381 IC50 = 50000 nM T07403 C1OS3A 12968382 IC50 = 122000 nM T07403 C8B9XH 12968383 IC50 = 60000 nM T07403 C8CHR1 12968384 IC50 = 85000 nM T07403 CWP8R7 12968385 IC50 = 82000 nM T07403 C5YOU2 12991693 IC50 = 16 nM T07403 CMNW32 16041071 IC50 = 62 nM T07403 C3IO0P 16122691 IC50 = 30 nM T07403 CXI61L 16122692 IC50 = 36 nM T07403 CGE4D6 16122706 IC50 = 29 nM T07403 C7SGL4 16122710 IC50 = 12 nM T07403 CLDK13 16678632 IC50 = 31 nM T07403 CJF3Z9 16678636 IC50 = 174 nM T07403 CSKE71 16678739 IC50 = 14 nM T07403 C9ZBU2 16678942 IC50 = 3 nM T07403 C3FZ4X 16678944 IC50 = 6 nM T07403 CB3QP4 16679038 IC50 = 50 nM T07403 C9JW4X 16679039 IC50 = 55 nM T07403 CN64QM 16679040 IC50 = 104 nM T07403 C3C4EA 16679140 IC50 = 4 nM T07403 CJ8R3B 16679443 IC50 = 12 nM T07403 CABL38 16679634 IC50 = 29 nM T07403 CYVJ37 16679722 IC50 = 67 nM T07403 CG3FV0 16727128 IC50 = 43 nM T07403 C9NHU3 20687429 IC50 = 89 nM T07403 C3DLN4 20793889 IC50 = 2100 nM T07403 C4NJ2L 20793895 IC50 = 2350 nM T07403 C1WN0S 20793908 IC50 = 62.5 nM T07403 C2D1UO 20793909 IC50 = 13 nM T07403 C1ZI3P 20793912 IC50 = 43.2 nM T07403 C27UDN 20793913 IC50 = 246 nM T07403 CVA8H3 20793914 IC50 = 58.6 nM T07403 CK0H4D 20793915 IC50 = 362 nM T07403 C3FW9R 20793916 IC50 = 299 nM T07403 C3W2BH 20793918 IC50 = 116 nM T07403 CF7TP9 20794038 IC50 = 166 nM T07403 C0Y1FH 21229395 IC50 = 1300 nM T07403 CVF32G 24748310 IC50 = 217 nM T07403 CR9EP2 24748311 IC50 = 510 nM T07403 C9NAX1 24748312 IC50 = 179 nM T07403 CE7P6Q 24748313 IC50 = 1368 nM T07403 C7UX2P 24748314 IC50 = 223 nM T07403 CWQ3H6 44277247 IC50 = 41 nM T07403 CLD1E0 44277294 IC50 = 1232 nM T07403 CIX4M7 44277304 IC50 = 53 nM T07403 C8HYQ2 44277327 IC50 = 306 nM T07403 CMN12S 44277340 IC50 = 160 nM T07403 CU4DX9 44277352 IC50 = 2.1 nM T07403 CL56IM 44277354 IC50 = 13 nM T07403 CA08RU 44277355 IC50 = 8.9 nM T07403 CSG1N6 44277413 IC50 = 197 nM T07403 C4V1MD 44284033 IC50 = 30000 nM T07403 CYK9Z6 44284064 IC50 = 117000 nM T07403 CYHI67 44284066 IC50 = 121000 nM T07403 CS47GU 44284171 IC50 = 16.3 nM T07403 CPH54Y 44284172 IC50 = 35.3 nM T07403 CO7Y3D 44284173 IC50 = 6.1 nM T07403 C0TC8Z 44284200 IC50 = 13.8 nM T07403 CZG56T 44284214 IC50 = 245 nM T07403 C6PW2K 44284215 IC50 = 22.3 nM T07403 CZI34O 44284227 IC50 = 16.1 nM T07403 CT0G2Q 44284229 IC50 = 26.6 nM T07403 CA48YS 44284230 IC50 = 19.6 nM T07403 CJ81ET 44284231 IC50 = 45.6 nM T07403 CT6C3W 44284239 IC50 = 275 nM T07403 CP4Y8X 44284243 IC50 = 11 nM T07403 CJB6G3 44284252 IC50 = 232 nM T07403 C0WH4U 44284316 IC50 = 504 nM T07403 CN0R8X 44284320 IC50 = 23.2 nM T07403 C3MSL9 44284375 IC50 = 176000 nM T07403 C6QJ8L 44284386 IC50 = 24.5 nM T07403 CSLM73 44284387 IC50 = 45.7 nM T07403 CZHQ16 44284392 IC50 = 8.49 nM T07403 C5S8QO 44284406 IC50 = 51.1 nM T07403 CWF83Z 44284417 IC50 = 99.5 nM T07403 CIQP20 44284419 IC50 = 327 nM T07403 C8BR4A 44284432 IC50 = 149 nM T07403 C52WLJ 44284486 IC50 = 733 nM T07403 C9SL1V 44284494 IC50 = 67 nM T07403 CMZ5O4 44284517 IC50 = 226.5 nM T07403 CI1PJ9 44284534 IC50 = 7.8 nM T07403 C9D4ON 44284536 IC50 = 56.4 nM T07403 CI29RA 44284552 IC50 = 80 nM T07403 C5KNA7 44284553 IC50 = 499 nM T07403 CR7T5I 44284566 IC50 = 22 nM T07403 C28RWG 44284602 IC50 = 374 nM T07403 C6E7CQ 44284627 IC50 = 11.24 nM T07403 CH7S9Z 44284643 IC50 = 22.95 nM T07403 CS8M0W 44284678 IC50 = 14.5 nM T07403 C3IL7K 44287646 IC50 = 465000 nM T07403 CU31NV 44288627 IC50 = 3.51 nM T07403 CI2C3Y 44288628 IC50 = 12.3 nM T07403 CQ48WG 44288629 IC50 = 62.4 nM T07403 CQG2B8 44288785 IC50 = 211 nM T07403 CV9Y2B 44288796 IC50 = 4.4 nM T07403 CAU49W 44288817 IC50 = 29.8 nM T07403 C6WKT1 44288845 IC50 = 5.26 nM T07403 C0BQ5O 44288950 IC50 = 51.4 nM T07403 CZ4NS3 44308036 IC50 = 215 nM T07403 CCL84F 44308037 IC50 = 33 nM T07403 C1PYH2 44308049 IC50 = 180 nM T07403 CSR43Y 44308070 IC50 = 165 nM T07403 C8CJ4Z 44308163 IC50 = 30 nM T07403 CNAO24 44308174 IC50 = 51 nM T07403 CHKS25 44308192 IC50 = 83 nM T07403 C2R7UB 44308204 IC50 = 15 nM T07403 CZJ2E0 44308205 IC50 = 49 nM T07403 C5L4VX 44308206 IC50 = 98 nM T07403 C62LKH 44308239 IC50 = 120 nM T07403 C5IXM2 44308403 IC50 = 18 nM T07403 CL9D2J 44308404 IC50 = 26 nM T07403 CXFC47 44308412 IC50 = 36.3 nM T07403 CV1TM5 44308416 IC50 = 22 nM T07403 CP2J7O 44308429 IC50 = 44 nM T07403 C9XCH7 44308491 IC50 = 94 nM T07403 C85FUQ 44308492 IC50 = 94 nM T07403 CWQI12 44308513 IC50 = 158 nM T07403 C40OWE 44308514 IC50 = 16.7 nM T07403 CE7LC4 44309967 IC50 = 5.8 nM T07403 C9HJ0O 44309968 IC50 = 18 nM T07403 CY6S2Q 44309985 IC50 = 45 nM T07403 CA8I7F 44309987 IC50 = 2.5 nM T07403 C6T4NH 44310021 IC50 = 18.8 nM T07403 C6B7YP 44310233 IC50 = 5 nM T07403 C5BGH0 44310255 IC50 = 3.5 nM T07403 C9BE3Y 44310286 IC50 = 21 nM T07403 C30PME 44310537 IC50 = 5.5 nM T07403 C9VOA3 44310538 IC50 = 17.1 nM T07403 CJEU74 44310553 IC50 = 110 nM T07403 CL8E2H 44310557 IC50 = 8.9 nM T07403 CFN64L 44314348 IC50 = 35 nM T07403 C5FC1O 44314395 IC50 = 4090 nM T07403 C9AIZ6 44314396 IC50 = 4.1 nM T07403 C6SD1G 44314397 IC50 = 2.2 nM T07403 CW10DI 44314409 IC50 = 120 nM T07403 C8SI3H 44314412 IC50 = 69 nM T07403 CXJ58C 44314413 IC50 = 35 nM T07403 C4JO7L 44314429 IC50 = 3.2 nM T07403 CBN9O7 44314430 IC50 = 105 nM T07403 C8F5RV 44314534 IC50 = 98 nM T07403 CIW4N3 44314551 IC50 = 1695 nM T07403 CF34ZY 44314636 IC50 = 5.5 nM T07403 C8XGA3 44314668 IC50 = 8400 nM T07403 CI6LT9 44314705 IC50 = 40 nM T07403 C9ABU8 44314711 IC50 = 22 nM T07403 C4UDX6 44314760 IC50 = 21 nM T07403 C4JY1Q 44314800 IC50 = 43 nM T07403 CZ0D7Q 44314815 IC50 = 78 nM T07403 CT24UI 44314816 IC50 = 65 nM T07403 C4Q0BY 44314831 IC50 = 78 nM T07403 CD37UY 44314908 IC50 = 3000 nM T07403 CGFK94 44320794 IC50 = 292000 nM T07403 C4TMH0 44321086 IC50 = 301000 nM T07403 CC3Y6H 44321087 IC50 = 163000 nM T07403 CF5MI3 44321138 IC50 = 317000 nM T07403 C5TR3K 44321139 IC50 = 308000 nM T07403 C5TSO8 44324472 IC50 = 97.1 nM T07403 CW4K2Z 44324473 IC50 = 78.25 nM T07403 C7H1TW 44324487 IC50 = 669.9 nM T07403 C2ULQ5 44324488 IC50 = 77 nM T07403 CP2B8I 44324517 IC50 = 13.2 nM T07403 CX9DS5 44324688 IC50 = 242 nM T07403 C7R5ZM 44324730 IC50 = 3551.1 nM T07403 CMS19Y 44324731 IC50 = 82.7 nM T07403 C3TQ9H 44324732 IC50 = 24.32 nM T07403 CW2G4X 44324735 IC50 = 1235 nM T07403 CQ53DR 44324768 IC50 = 948.8 nM T07403 C50RSE 44324774 IC50 = 5720 nM T07403 C16XST 44324776 IC50 = 311 nM T07403 C4NK8T 44324794 IC50 = 413 nM T07403 C03KOG 44324807 IC50 = 52.5 nM T07403 CWG84B 44324812 IC50 = 1140.8 nM T07403 CJN8B3 44324819 IC50 > 4000 nM T07403 C2OJI4 44324820 IC50 = 344.5 nM T07403 COIG83 44324854 IC50 = 2260 nM T07403 CE3TH4 44330475 IC50 = 25 nM T07403 CL6RA9 44330517 IC50 = 53 nM T07403 CBME25 44330518 IC50 = 240 nM T07403 C4BJK6 44330548 IC50 = 50.3 nM T07403 CN0S7M 44330565 IC50 = 47.7 nM T07403 CA3UX5 44330581 IC50 = 10 nM T07403 C13PBU 44330595 IC50 = 22 nM T07403 CXTA89 44330626 IC50 = 11.3 nM T07403 CWN4L8 44330629 IC50 = 12 nM T07403 CJ4E6H 44330660 IC50 = 736 nM T07403 CX46NY 44343237 IC50 = 30 nM T07403 CF38BE 44343238 IC50 = 260 nM T07403 CFQ6R5 44343239 IC50 = 340 nM T07403 C8L4HI 44343263 IC50 = 110 nM T07403 CU5Z9G 44343282 IC50 = 2200 nM T07403 C6AJ8U 44343283 IC50 = 20000 nM T07403 C80DNY 44343284 IC50 = 2100 nM T07403 C5A0BF 44343310 IC50 = 190 nM T07403 CHP40V 44343311 IC50 = 640 nM T07403 CFX5B7 44343326 IC50 > 100000 nM T07403 CNMQ48 44343327 IC50 = 2200 nM T07403 C9E8NP 44343328 IC50 = 1100 nM T07403 CV9M6T 44343453 IC50 = 520 nM T07403 CL8E3T 44343454 IC50 = 550 nM T07403 COM1C6 44343455 IC50 = 130 nM T07403 CQ8Z1H 44343585 IC50 = 120 nM T07403 CU0A2D 44343587 IC50 = 40000 nM T07403 CW97VR 44343589 IC50 = 840 nM T07403 CHX5I8 44343599 IC50 = 40000 nM T07403 C53TVL 44343600 IC50 = 130 nM T07403 CHF18Y 44343602 IC50 = 11000 nM T07403 C0LGN6 44343603 IC50 = 4500 nM T07403 CO12WD 44343604 IC50 = 1800 nM T07403 CO7R5Y 44343621 IC50 > 100000 nM T07403 C35FPB 44343634 IC50 = 290 nM T07403 C19TDW 44343641 IC50 = 250 nM T07403 CPZE98 44343642 IC50 = 23000 nM T07403 CJ73KU 44343656 IC50 = 30000 nM T07403 CHQ96V 44343657 IC50 = 175000 nM T07403 C6K8DG 44343677 IC50 = 10000 nM T07403 CC35LO 44343703 IC50 = 1900 nM T07403 C0I9YS 44343704 IC50 = 390 nM T07403 CRUH62 44343705 IC50 = 430 nM T07403 C4UJW3 44372342 IC50 = 2850 nM T07403 C1GDE4 44382099 IC50 = 91 nM T07403 C8UG4P 44382103 IC50 = 83 nM T07403 CDO7I6 44382111 IC50 = 58 nM T07403 CY40TS 44382171 IC50 = 388 nM T07403 CK2GI4 44382174 IC50 = 52 nM T07403 C6MEZ0 44382232 IC50 = 19 nM T07403 C6AO0T 44382423 IC50 = 20 nM T07403 CY2C6E 44382469 IC50 = 179 nM T07403 CPSO78 44382497 IC50 = 5.2 nM T07403 CO5FU2 44382554 IC50 = 70 nM T07403 CNFM87 44382556 IC50 = 318 nM T07403 CIEX15 44382584 IC50 = 150 nM T07403 CQHD50 44382635 IC50 = 38 nM T07403 C0RL7W 44382645 IC50 = 7335 nM T07403 C05FRE 44382649 IC50 = 3.2 nM T07403 CGMN67 44382676 IC50 = 45 nM T07403 CAR47D 44382683 IC50 = 13 nM T07403 C28BMU 44382684 IC50 = 5 nM T07403 C0AY8L 44382685 IC50 = 54 nM T07403 C45QUC 44382714 IC50 = 5 nM T07403 C6TLQ9 44382715 IC50 = 40 nM T07403 C91HRV 44382716 IC50 = 53 nM T07403 C1OP9Q 44382723 IC50 = 149 nM T07403 CLMI61 44382729 IC50 = 25 nM T07403 CDK46W 44382769 IC50 = 521 nM T07403 CRL9V3 44382770 IC50 = 4 nM T07403 C0BR5U 44382771 IC50 = 147 nM T07403 C1QF5Y 44382777 IC50 = 5 nM T07403 CSIT45 44382810 IC50 = 77 nM T07403 C7L5TE 44382824 IC50 = 128 nM T07403 CL2G1B 44382830 IC50 = 16 nM T07403 C9SQ6Y 44387471 IC50 = 17 nM T07403 CJ9H5K 44430327 IC50 = 13000 nM T07403 C5F4KM 44454106 IC50 = 8600 nM T07403 CA3F9K 44454449 IC50 = 1600 nM T07403 CPU15F 44454450 IC50 = 180 nM T07403 CO4YE7 44454480 IC50 = 36 nM T07403 C1ZNQ8 44454481 IC50 = 39 nM T07403 C3AGH7 44454515 IC50 = 24 nM T07403 CI1A9S 44454544 IC50 = 21 nM T07403 C3IW1E 44454549 IC50 = 69 nM T07403 CDW2G9 44454578 IC50 = 25 nM T07403 CS81QU 44454580 IC50 = 13 nM T07403 C72NXQ 44454604 IC50 = 19 nM T07403 CN2D6B 44454606 IC50 = 23 nM T07403 CFY48V 44454634 IC50 = 61 nM T07403 CK5EN8 44454635 IC50 = 21 nM T07403 CW5SF4 44454656 IC50 = 78 nM T07403 C5WF3A 44454658 IC50 = 89 nM T07403 CIU9A7 44454686 IC50 = 230 nM T07403 C5OZ7S 44454712 IC50 = 80 nM T07403 CCPW89 44454736 IC50 = 35 nM T07403 CX0N7J 44454738 IC50 = 18 nM T07403 CLA4C0 51346866 IC50 = 510 nM T07403 CD8KJ6 54686083 IC50 = 49 nM T07403 C2L7DX 56671702 IC50 > 100000 nM T07403 CDU79K 56678432 IC50 = 43000 nM T07403 C8UQ4J 56681774 IC50 = 7900 nM T07403 CA82IB 69232792 IC50 = 671 nM T07403 C9QZG0 69335939 IC50 = 219 nM T07403 CSC75B 69335964 IC50 = 58 nM T07403 CSOG60 69336100 IC50 = 124 nM T07403 C6I8MK 69336784 IC50 = 151 nM T07403 CZEN52 69336954 IC50 = 167 nM T07403 C2SDK6 69337248 IC50 = 35 nM T07403 CO2M1D 69337579 IC50 = 81 nM T07403 C28KZD 69714759 IC50 = 767 nM T07403 CFU54E 69714767 IC50 = 154 nM T07403 CK5C3Q 69715313 IC50 = 126 nM T07403 CP5Y8I 69715941 IC50 = 160 nM T07403 C0G7XN 69716544 IC50 = 1290 nM T07403 C76YRK 71552171 IC50 = 810 nM T07403 C60QOE 71552172 IC50 = 61 nM T07403 C6YE4B 71552173 IC50 = 1230 nM T07403 C4OT8U 71553149 IC50 = 558 nM T07403 C6YS7E 71716980 IC50 = 600 nM T07403 C4HY2C 71717599 IC50 = 1970 nM T07403 CY13HN 71720011 IC50 = 254 nM T07403 CS0D7R 71727849 IC50 = 419 nM T07403 C6QJA2 71727850 IC50 = 4549 nM T07403 CD1NH6 71727851 IC50 = 311 nM T07403 C1B7MR 71727976 IC50 = 3002 nM T07403 CEG34M 71727977 IC50 = 156 nM T07403 CU5CB6 71727978 IC50 = 321 nM T07403 CW6T4H 71728104 IC50 = 262 nM T07403 CMC5Q3 71728105 IC50 = 483 nM T07403 CN3QT4 71728106 IC50 = 1054 nM T07403 CQ8HY9 71728107 IC50 = 468 nM T07403 C59QKD 71728220 IC50 = 594 nM T07403 CB95ZS 71728221 IC50 = 151 nM T07403 C9R1BP 71728222 IC50 = 3684 nM T07403 CV7DK0 122181680 IC50 = 270 nM T07403 CWY3V2 122181682 IC50 = 343 nM T07403 CPU86F 135438774 IC50 = 60 nM T07403 CIJ2F3 135451177 IC50 > 20000 nM T07403 C9ONY2 135458887 IC50 = 900 nM T07403 CWKN67 135614554 IC50 = 10000 nM T07403 C3JVT0 136152923 IC50 = 260 nM T07403 CM6YS7 136152928 IC50 = 5500 nM T07403 D0A0JM 10120218 EC50 = 1.4 nM T51120 D00MIN 657298 IC50 = 3380 nM T51120 D0Y3LJ 10264211 IC50 = 3900 nM T51120 CBC0J5 6418797 IC50 > 30000 nM T51120 CC9S5U 28412206 IC50 = 6000 nM T51120 C5MQR9 130365202 IC50 = 4000 nM T52382 C2WNO3 145957990 IC50 = 9080 nM T52382 CPC30D 145958830 IC50 = 6830 nM T52382 C2ZI8C 145973614 IC50 = 4220 nM T82702 D01AQT 441383 EC50 = 8900 nM T82702 D01VMO 3401 EC50 = 6100 nM T82702 D01XBA 5035 EC50 = 11710 nM T82702 D02HWP 2722 EC50 = 39800 nM T82702 D02LZB 220401 EC50 = 12600 nM T82702 D04ITO 6436173 EC50 = 2200 nM T82702 D05DVP 5717 EC50 = 710 nM T82702 D06ABF 3957 EC50 = 3000 nM T82702 D06OMK 445643 EC50 = 5000 nM T82702 D06RGG 5819 EC50 = 11200 nM T82702 D06ZAY 3561 EC50 = 10000 nM T82702 D08PIQ 6741 EC50 = 12600 nM T82702 D0AJ5L 4615 EC50 = 400 nM T82702 D0CZ1Q 5311067 EC50 = 31600 nM T82702 D0D2TN 5311412 EC50 = 400 nM T82702 D0E1WI 3345 EC50 = 31600 nM T82702 D0E7PQ 5311 EC50 = 25100 nM T82702 D0G3DL 135398735 EC50 = 190 nM T82702 D0G8BV 6450278 IC50 = 2.4 nM T82702 D0I3RO 92974 EC50 = 4 nM T82702 D0JO7Y 104741 EC50 = 1950 nM T82702 D0P0HT 9878 EC50 = 1300 nM T82702 D0P1FO 16078 EC50 = 12600 nM T82702 D0S5CU 4499 EC50 = 7900 nM T82702 D0T9TJ 3034010 EC50 = 1600 nM T82702 D0U4CE 104865 EC50 = 8900 nM T82702 D0WN0U 3333 EC50 = 1900 nM T82702 D0X2IE 3080 EC50 = 5000 nM T82702 D0X5ZI 6918493 EC50 = 31600 nM T82702 D0Y2NE 448537 IC50 = 14600 nM T82702 D0ZU9R 392622 EC50 = 4000 nM T82702 D00WDY 53477157 EC50 > 50000 nM T82702 D02EVF 6112 EC50 = 2800 nM T82702 D04TNT 46851313 EC50 > 10000 nM T82702 D06GRK 4494 EC50 = 890 nM T82702 D08SCL 46190695 EC50 > 30000 nM T82702 D0B5HF 44476893 EC50 > 10000 nM T82702 D0DH5X 44472635 EC50 > 30000 nM T82702 D0DK8X 50922691 EC50 > 50000 nM T82702 D0H2UB 5361 EC50 = 1300 nM T82702 D0H4DR 49787490 EC50 = 1000 nM T82702 D0H7QU 56934415 EC50 > 50000 nM T82702 D0I3TU 45268455 EC50 > 30000 nM T82702 D0LQ3L 77108121 EC50 = 13000 nM T82702 D0S2PD 42634627 EC50 > 50000 nM T82702 D0UX2V 44537841 EC50 > 25000 nM T82702 D0W1US 1684 EC50 = 251.19 nM T82702 D0W1XE 91827457 IC50 > 10000 nM T82702 D0YZ8I 4273754 EC50 = 2640 nM T82702 D0C7RV 446313 EC50 = 80 nM T82702 D0CV7Z 448013 EC50 = 12600 nM T82702 D0F8IO 5773 EC50 = 3200 nM T82702 D0H7WA 60496 EC50 = 28200 nM T82702 D0QQ1J 2406 EC50 = 1000 nM T82702 D0Y7VM 47936 EC50 = 700 nM T82702 C25CAT 122184111 EC50 = 9900 nM T82702 CYDS15 3326 EC50 = 1300 nM T82702 CY2F4Q 3334 EC50 = 10000 nM T82702 C2NX4F 11102 EC50 = 11200 nM T82702 CN63MS 42725 EC50 = 28200 nM T82702 CJ7M5B 65341 EC50 = 12600 nM T82702 C9I4OL 65770 EC50 = 1100 nM T82702 CMH80E 68909 EC50 = 1600 nM T82702 CQ65YS 92112 EC50 = 12600 nM T82702 CD34EB 122081 EC50 = 3200 nM T82702 CA34IS 231084 EC50 = 11200 nM T82702 C7VUP3 421450 EC50 = 271 nM T82702 C3J2LX 456389 EC50 = 7900 nM T82702 CG93IP 1475852 EC50 > 50000 nM T82702 C50GWH 1550998 EC50 = 10000 nM T82702 CLAM57 2744646 IC50 = 850 nM T82702 C8G1OD 2746124 IC50 = 850 nM T82702 CHJ15W 2837530 EC50 = 3500 nM T82702 CXL52Q 2961516 EC50 = 49 nM T82702 CJ6Z8I 2999413 EC50 = 4000 nM T82702 CA6WB3 3032539 EC50 = 10500 nM T82702 CY5F7Z 5377791 EC50 = 7900 nM T82702 CB83IO 5462355 EC50 = 14100 nM T82702 C46NFC 6426773 EC50 = 5600 nM T82702 C4UCM5 6434217 EC50 = 5000 nM T82702 C16ZSG 6439929 IC50 = 2.4 nM T82702 CBV1E2 9568628 EC50 = 25100 nM T82702 CJDP76 9838675 EC50 = 30000 nM T82702 CGEJ24 9985625 EC50 > 25000 nM T82702 CG0LQ8 10129170 Ki > 10000 nM T82702 CF9PG8 10218693 Ki > 10000 nM T82702 C7IUQ6 10335880 EC50 = 1600 nM T82702 CI64PJ 10340916 EC50 = 1700 nM T82702 C6UJ4O 10455173 EC50 = 1300 nM T82702 CP53LK 11583743 IC50 > 10000 nM T82702 C31MCZ 11957704 EC50 = 7100 nM T82702 C3N7VE 15953424 EC50 = 150 nM T82702 CEYW48 15953464 EC50 > 50000 nM T82702 C7UCS5 16064456 EC50 = 3300 nM T82702 C0V9RI 16064896 EC50 > 30000 nM T82702 C4UB6X 16064899 EC50 > 30000 nM T82702 CN89BT 16065038 EC50 > 30000 nM T82702 C2VH9W 16065039 EC50 > 30000 nM T82702 C4KNH5 16065040 EC50 > 30000 nM T82702 CL0KD4 16065041 EC50 > 30000 nM T82702 CO93MX 16065042 EC50 > 30000 nM T82702 C0DVS7 16072077 EC50 = 3.162 nM T82702 CHX0Z8 16117661 EC50 > 50000 nM T82702 C0CRS4 16663280 IC50 = 4800 nM T82702 CPVC43 16749938 EC50 > 30000 nM T82702 CC09QT 16759171 EC50 = 4000 nM T82702 CH4MZ2 17757343 EC50 > 50000 nM T82702 C2LMW1 18565134 EC50 = 940 nM T82702 C0QKH8 18565138 EC50 = 1100 nM T82702 CGS1R9 18565141 EC50 = 820 nM T82702 C38JEL 20704150 EC50 = 39 nM T82702 C3GY4C 23641891 EC50 = 4300 nM T82702 C9WSK4 23642165 EC50 = 430 nM T82702 CI7W3Z 23642174 EC50 = 5000 nM T82702 CMS87Z 23650702 EC50 > 50000 nM T82702 CMG9P7 23652708 EC50 > 50000 nM T82702 C60OSF 23652709 EC50 > 50000 nM T82702 C4O9IX 23652854 EC50 > 50000 nM T82702 CYTN73 23652855 EC50 > 50000 nM T82702 C13UFH 23652857 EC50 > 50000 nM T82702 COL1N6 23652916 EC50 > 50000 nM T82702 C1MB8K 23663953 EC50 = 14100 nM T82702 CV7GX0 23672302 EC50 = 6300 nM T82702 C0OBD9 23677058 EC50 = 4100 nM T82702 CXH32E 23678597 EC50 = 6300 nM T82702 CUS67W 23707968 EC50 = 15800 nM T82702 CDS4T7 24744018 EC50 > 50000 nM T82702 CTE1N2 24748569 EC50 > 1282000 nM T82702 C57DJQ 24750734 IC50 > 25000 nM T82702 C3S8NH 24752568 IC50 > 25000 nM T82702 C3P7IS 24768572 IC50 > 30000 nM T82702 C8N1RD 24776331 EC50 = 1000 nM T82702 C1U5CP 24776332 EC50 = 501.19 nM T82702 C4W1LF 24776334 EC50 = 158.49 nM T82702 C38CHU 24776335 IC50 = 7943.28 nM T82702 CTXB68 24776336 EC50 = 10000 nM T82702 C0TYF8 24776337 EC50 = 10000 nM T82702 CS0YZ8 24776338 EC50 = 15.85 nM T82702 C0Z2OY 24776339 IC50 = 630.96 nM T82702 C59ZYO 24776340 EC50 = 10 nM T82702 CQHV30 24857855 EC50 = 1700 nM T82702 CI81ZP 24945724 EC50 > 50000 nM T82702 CK5TJ7 24945801 EC50 > 50000 nM T82702 C9ZY2N 25016295 EC50 = 1000 nM T82702 CXJ3N9 25018323 EC50 = 9000 nM T82702 CZ3RK7 25018324 EC50 > 50000 nM T82702 CZVG24 25019000 EC50 > 50000 nM T82702 C5UNW6 25019002 EC50 = 3000 nM T82702 CYJ9W8 25024037 EC50 = 600 nM T82702 CNW89T 25026445 EC50 > 25000 nM T82702 CIC1G3 25100139 EC50 = 6640 nM T82702 CM8TL0 25100141 EC50 = 570 nM T82702 CBIJ72 25101376 EC50 > 30000 nM T82702 CPZ4A8 25101678 EC50 = 1810 nM T82702 CL8B4H 25101818 EC50 > 30000 nM T82702 CUYI02 25101821 EC50 > 30000 nM T82702 C1FN2Y 25101822 EC50 > 30000 nM T82702 CR6F2B 25102111 EC50 > 30000 nM T82702 C82HQP 25102249 EC50 = 10760 nM T82702 C78RUM 25134006 EC50 > 30000 nM T82702 CQHC91 25134007 EC50 = 2400 nM T82702 CUX49Z 25144536 EC50 > 50000 nM T82702 C53PTZ 25256089 EC50 > 30000 nM T82702 CA4GR8 25256749 EC50 = 6000 nM T82702 CA25BL 42603033 EC50 > 30000 nM T82702 CE0G6W 42633574 EC50 > 50000 nM T82702 CYC3O1 42634126 EC50 > 50000 nM T82702 CK79IO 42634797 EC50 = 25000 nM T82702 C9R7PZ 42634800 EC50 = 25000 nM T82702 CX7D8M 42634801 EC50 = 48000 nM T82702 CID91J 42634802 EC50 = 3600 nM T82702 CAS1M0 44428685 EC50 = 125.89 nM T82702 CR5SI0 44476535 EC50 = 3871000 nM T82702 CV09AF 44567313 EC50 = 20 nM T82702 C0BNS1 44567314 EC50 = 176 nM T82702 C69FLG 44567315 EC50 = 428 nM T82702 CC0KU9 44567319 EC50 = 23 nM T82702 CL6TR0 44567320 EC50 = 376 nM T82702 C3I7VQ 44567321 EC50 = 340 nM T82702 CE4AU0 44567322 EC50 = 197 nM T82702 CXZ06J 44567323 EC50 = 1456 nM T82702 CH6R7S 44567331 EC50 > 5000 nM T82702 CH42CP 44567332 EC50 = 388 nM T82702 C0Y3SK 44567333 EC50 = 45 nM T82702 C2R4EW 44567334 EC50 = 33 nM T82702 C8MQ4W 44567335 EC50 = 1.5 nM T82702 CUEQ15 44567342 EC50 > 5000 nM T82702 C6BUF4 44567343 EC50 = 515 nM T82702 CPT34X 44567344 EC50 = 217 nM T82702 CIJ89X 44567345 EC50 > 5000 nM T82702 C01GYR 44567346 EC50 = 20 nM T82702 CV9C1X 44567354 EC50 = 0.7 nM T82702 CA76WD 44567355 EC50 = 42 nM T82702 CK1W6C 44567356 EC50 = 52 nM T82702 C6D8QY 44567357 EC50 = 55 nM T82702 C7RH1O 44567358 EC50 = 13 nM T82702 CQ7J0V 44567365 EC50 = 101 nM T82702 C3ZQY7 44567366 EC50 = 271 nM T82702 C83KUY 44567367 EC50 = 336 nM T82702 CY6DC4 44567368 EC50 = 51 nM T82702 C8OXL3 44567374 EC50 = 385 nM T82702 CPB36X 44567375 EC50 = 55 nM T82702 CO5YU9 44576846 EC50 = 3600 nM T82702 CV6I1C 44576848 EC50 = 7700 nM T82702 C9TC4U 44576849 EC50 = 1700 nM T82702 C6ZU1A 44576872 EC50 = 2400 nM T82702 C4YIR7 44576873 EC50 > 25000 nM T82702 CRA54F 44576874 EC50 = 12000 nM T82702 C2HW0I 44576875 EC50 > 25000 nM T82702 C51WSL 44576899 EC50 > 25000 nM T82702 CF2B1H 44576901 EC50 = 1300 nM T82702 C0JH2G 44576902 EC50 = 3200 nM T82702 CWRD09 44576943 EC50 = 7900 nM T82702 CWX1Z0 44576944 EC50 > 25000 nM T82702 COQ7U4 44576945 EC50 = 700 nM T82702 C6P5ER 44576967 EC50 = 25000 nM T82702 C4IY8M 45256689 EC50 > 30000 nM T82702 C7CK6V 46178246 EC50 > 50000 nM T82702 CRF6X8 46887882 EC50 > 30000 nM T82702 CJ3FM4 46925833 EC50 > 3000 nM T82702 CJK53D 46933697 IC50 > 25000 nM T82702 CZ0G6A 46947062 IC50 = 8400 nM T82702 C2D6PB 49771960 EC50 > 3000 nM T82702 CWU2R3 49773361 EC50 > 50000 nM T82702 CM3ZF5 49779868 EC50 = 3300 nM T82702 CG6LI3 49822225 EC50 = 3000 nM T82702 CU63QR 49847377 IC50 > 30000 nM T82702 CJ7H2B 49847753 IC50 > 50000 nM T82702 C05SEW 49849008 IC50 > 30000 nM T82702 C78SAD 49849115 IC50 > 50000 nM T82702 CUD91T 49862248 EC50 = 390000 nM T82702 CENW12 50925404 IC50 > 25000 nM T82702 CFD09E 50925451 EC50 = 5200 nM T82702 C42BOI 52942803 IC50 > 25000 nM T82702 CM36DN 52943994 IC50 > 25000 nM T82702 CQ0RX5 52945526 EC50 = 15800 nM T82702 CA3UB6 52947647 IC50 > 25000 nM T82702 C6LSO0 52948590 IC50 > 25000 nM T82702 C74IUF 52948931 IC50 = 3300 nM T82702 C3VMQ5 52949827 IC50 = 4500 nM T82702 CXV3W2 53317718 EC50 > 30000 nM T82702 CP14EK 53317957 EC50 > 30000 nM T82702 C2NH0C 53319296 EC50 > 30000 nM T82702 COJ82D 53319320 EC50 > 30000 nM T82702 CD79XG 53321898 EC50 = 740 nM T82702 C1H7AG 53323238 EC50 = 600 nM T82702 CN83JY 53325880 EC50 = 940 nM T82702 CZ1SE0 53325908 EC50 > 30000 nM T82702 C8PJ6E 53354789 EC50 = 3000 nM T82702 C7I8YR 53465062 EC50 = 1300 nM T82702 CN93FS 54580118 EC50 > 30000 nM T82702 CF05VK 54580143 EC50 > 30000 nM T82702 C7FXV6 54580144 EC50 > 30000 nM T82702 CBX17R 54581094 EC50 > 30000 nM T82702 C8O9WK 54581095 EC50 > 30000 nM T82702 CM67RK 54581096 EC50 > 30000 nM T82702 C8ZDF3 54581137 EC50 > 30000 nM T82702 CQ7GV2 54582134 EC50 > 30000 nM T82702 CZ1B6L 54582135 EC50 > 30000 nM T82702 C07KDH 54582136 EC50 > 30000 nM T82702 CK29GC 54582137 EC50 > 30000 nM T82702 CKGX19 54582164 EC50 > 30000 nM T82702 CM2QX4 54583079 EC50 > 30000 nM T82702 CMKQ26 54583080 EC50 > 30000 nM T82702 C2G7LK 54583125 EC50 > 30000 nM T82702 CL6Z9X 54583126 EC50 > 30000 nM T82702 CGM2W4 54583127 EC50 > 30000 nM T82702 CF42QY 54583128 EC50 > 30000 nM T82702 CZ4YV3 54584081 EC50 > 30000 nM T82702 CHP62C 54584119 EC50 > 30000 nM T82702 CD2QO1 54584120 EC50 = 3000 nM T82702 CCT0B2 54584121 EC50 = 4800 nM T82702 C0VPS6 54584122 EC50 > 30000 nM T82702 CGD4N3 54585028 EC50 > 30000 nM T82702 C8NZ2B 54585029 EC50 > 30000 nM T82702 CHW48S 54585030 EC50 > 30000 nM T82702 CZ8R0S 54585053 EC50 > 30000 nM T82702 C04IZR 54585054 EC50 > 30000 nM T82702 C5SHO2 54585992 EC50 > 30000 nM T82702 CJA5Z6 54585993 EC50 > 30000 nM T82702 C4JTZ5 54585994 EC50 = 8700 nM T82702 CKF15E 54586030 EC50 > 30000 nM T82702 CT12RX 54586031 EC50 = 23000 nM T82702 CJ8K1Y 54586966 EC50 > 30000 nM T82702 C51MDN 54586967 EC50 = 18000 nM T82702 CH2F8P 54586968 EC50 > 30000 nM T82702 C61ZTA 54586969 EC50 > 30000 nM T82702 C3Y6HF 54587012 EC50 = 4600 nM T82702 CXU62W 54677935 EC50 > 50000 nM T82702 C67LSP 54685047 EC50 = 3200 nM T82702 C28RDF 54746913 EC50 > 30000 nM T82702 C69EQM 54752774 EC50 = 31622.78 nM T82702 C91PGO 56603115 IC50 > 30000 nM T82702 C5ES6P 56603116 IC50 > 30000 nM T82702 CVI51O 56603118 IC50 > 30000 nM T82702 C2IM6T 56603174 IC50 > 30000 nM T82702 CH05TN 56603175 IC50 > 30000 nM T82702 CDL94H 56603301 IC50 > 30000 nM T82702 C9D1MV 56603353 IC50 > 30000 nM T82702 CDS9Y3 56659419 EC50 = 150 nM T82702 C6RU0N 56659420 EC50 = 150 nM T82702 CI54DZ 56676581 EC50 = 150 nM T82702 CF1O6J 56679929 EC50 = 150 nM T82702 CQ4H9K 56683246 EC50 = 150 nM T82702 C3NPO1 56683248 EC50 = 150 nM T82702 CFO23H 56837193 EC50 = 260 nM T82702 C71JRF 56949451 EC50 = 2300 nM T82702 CP6AS2 56952795 EC50 > 250000 nM T82702 C1AV7C 56970444 EC50 = 2460 nM T82702 C9S8MU 57386524 IC50 > 50000 nM T82702 C3N4MF 57520842 EC50 > 30000 nM T82702 CEL56T 57520942 EC50 > 30000 nM T82702 C7VF2J 57550042 EC50 > 50000 nM T82702 C7BDI5 57580339 EC50 = 8400 nM T82702 CN7YT4 57652306 EC50 = 1300 nM T82702 C35GXV 57720515 EC50 > 50000 nM T82702 C8A5FH 57720601 EC50 > 50000 nM T82702 CJ17LO 57808861 EC50 = 970 nM T82702 C3XQZ4 57808870 EC50 = 500 nM T82702 C0GN3C 57808912 EC50 = 300 nM T82702 CK3E2N 57808982 EC50 = 1200 nM T82702 CL38KT 57808983 EC50 = 2600 nM T82702 CRDS36 57808989 EC50 = 400 nM T82702 C39YAD 57809000 EC50 = 1100 nM T82702 C05XBJ 57809011 EC50 = 2800 nM T82702 CCFD09 57809042 EC50 = 800 nM T82702 CUG73D 57888785 EC50 = 19000 nM T82702 CP13VI 57889180 EC50 > 50000 nM T82702 CMZQ02 57889181 EC50 = 1800 nM T82702 C31ZKO 57889736 EC50 = 5700 nM T82702 CLH4Y8 57991707 EC50 = 1400 nM T82702 CWXC70 58180596 EC50 > 16000 nM T82702 CCQM76 59153288 EC50 > 30000 nM T82702 C9VNB7 59275242 EC50 = 1600 nM T82702 CTF1U6 59275404 EC50 > 50000 nM T82702 CTVM01 59337052 EC50 > 50000 nM T82702 C6E5DX 59337191 EC50 = 6700 nM T82702 CG5QX1 59337199 EC50 > 50000 nM T82702 CXO18I 59337218 EC50 > 25000 nM T82702 CPUZ69 59447115 EC50 = 2500 nM T82702 CXH19J 59472574 EC50 > 30000 nM T82702 CAKY62 59618747 EC50 = 1800 nM T82702 C8UJ7N 59618753 EC50 = 3500 nM T82702 CEU67L 59618790 EC50 > 10000 nM T82702 CWR3U0 62707207 EC50 = 10000 nM T82702 CV4BD2 62707362 EC50 = 1100 nM T82702 CYU24M 62707363 EC50 = 6600 nM T82702 CXD5M1 62707364 EC50 = 11800 nM T82702 C8SKU9 62707365 EC50 > 10000 nM T82702 C2E0YG 62707528 EC50 > 25000 nM T82702 C2LBW7 66551925 EC50 > 30000 nM T82702 CBOF40 68046989 IC50 > 30000 nM T82702 C1XHA8 71116039 IC50 > 30000 nM T82702 C32UMV 71203748 IC50 > 30000 nM T82702 C6BE5X 71271461 EC50 > 30000 nM T82702 CH1S3G 71548918 EC50 = 16700 nM T82702 CT4G9E 71555441 EC50 = 5700 nM T82702 C1DR8E 71622396 EC50 = 3000 nM T82702 C86DGB 71681399 EC50 = 8500 nM T82702 CTX46Q 71770951 EC50 > 50000 nM T82702 C7B6JU 72543966 EC50 = 2700 nM T82702 CMZ85K 72722807 EC50 = 571 nM T82702 C2BQO3 72722945 EC50 = 190 nM T82702 CH1JK9 73213123 EC50 > 50000 nM T82702 C34DYM 74369475 EC50 > 50000 nM T82702 C0ATV1 74369476 EC50 > 50000 nM T82702 C6UWO5 74762670 EC50 > 10000 nM T82702 CPS18J 75276948 EC50 = 2000 nM T82702 CJXG25 76284182 EC50 > 10000 nM T82702 CZX32H 76310864 EC50 = 21000 nM T82702 C3ZQU4 76310996 EC50 > 50000 nM T82702 C02XJO 76313667 EC50 = 1900 nM T82702 CK91LZ 76314629 EC50 > 50000 nM T82702 CNY2D6 76321910 EC50 > 50000 nM T82702 CQN91E 76324551 EC50 = 10800 nM T82702 CZYW47 76328940 EC50 = 18000 nM T82702 CWD5R4 76331595 EC50 > 15000 nM T82702 CWJ65U 76331788 EC50 = 2800 nM T82702 C9CTQ0 76331789 EC50 = 1700 nM T82702 C4OXA6 76331790 EC50 > 10000 nM T82702 CV6KW2 76335376 EC50 = 6800 nM T82702 CGE5S3 76336366 EC50 > 50000 nM T82702 CRY6D5 76336383 EC50 > 50000 nM T82702 C8CP3K 76903477 EC50 > 25000 nM T82702 C34TAM 77845572 EC50 > 30000 nM T82702 C2NCH9 78318214 EC50 > 30000 nM T82702 C2GET7 78318815 EC50 > 30000 nM T82702 CBI06J 86346645 EC50 > 10000 nM T82702 C5VCM4 86690644 EC50 > 10000 nM T82702 CGFW70 86690646 EC50 > 10000 nM T82702 CC8I0M 86707711 EC50 > 17000 nM T82702 CTW8L6 86766622 EC50 = 5600 nM T82702 CR0P6K 89584034 EC50 > 30000 nM T82702 C5MOV2 89659415 EC50 > 10000 nM T82702 C7E5RV 90200534 EC50 > 10000 nM T82702 C26LKW 90341025 EC50 > 30000 nM T82702 C02PKF 90644224 IC50 = 11000 nM T82702 C2M0NE 90644225 IC50 = 14000 nM T82702 C9QZE2 91039859 EC50 = 1000 nM T82702 CI92WR 91664317 EC50 > 10000 nM T82702 C9ETC1 91666645 EC50 = 5600 nM T82702 C60HAJ 91885643 EC50 = 19000 nM T82702 CT3K8B 117940657 EC50 = 2000 nM T82702 C9R5HF 117949985 EC50 = 2000 nM T82702 C0W6MZ 117950226 EC50 = 1100 nM T82702 C4S9EM 117964962 EC50 > 10000 nM T82702 CS4GJ9 117964973 EC50 > 10000 nM T82702 CDXK37 117964975 EC50 > 10000 nM T82702 CN6RT8 117964978 EC50 > 10000 nM T82702 C96BSK 117964998 EC50 > 10000 nM T82702 CW27MY 118063735 EC50 > 30000 nM T82702 CMX3U8 118107483 EC50 > 5480 nM T82702 CWR6I1 118112300 EC50 = 16000 nM T82702 C79IOD 118207841 EC50 > 50000 nM T82702 CW27ZE 118207854 EC50 > 50000 nM T82702 CXW5M0 118207954 EC50 > 50000 nM T82702 C9UK5A 118207966 EC50 = 1800 nM T82702 C0SQH5 118207970 EC50 = 4930 nM T82702 C0PWH6 118207991 EC50 > 50000 nM T82702 C2U3TJ 118208018 EC50 > 50000 nM T82702 C1MOT7 118208026 EC50 = 6440 nM T82702 CZ2C3U 118208048 EC50 > 18000 nM T82702 CI86YW 118208079 EC50 = 434 nM T82702 C2KAR6 118208086 EC50 = 12600 nM T82702 C3TJY2 118208092 EC50 = 520 nM T82702 CS2F1K 118208112 EC50 = 7810 nM T82702 C8N2PF 118208184 EC50 > 50000 nM T82702 C9GU8A 118212056 EC50 = 239 nM T82702 CWO9G0 118212096 EC50 = 10 nM T82702 CKW6P1 118212175 EC50 = 752 nM T82702 CEU56B 118212311 EC50 = 1010 nM T82702 CKU79R 118212564 EC50 = 275 nM T82702 C4DRH0 118212615 EC50 = 229 nM T82702 C51XTL 118217548 EC50 = 794 nM T82702 C1FL5I 118217550 EC50 = 480 nM T82702 CEN76C 118217555 EC50 > 2470 nM T82702 CH9T1O 118217580 EC50 > 5140 nM T82702 CIT31Q 118217593 EC50 > 50000 nM T82702 C1ZRN9 118217594 EC50 > 50000 nM T82702 CAUT58 118217595 EC50 > 50000 nM T82702 CB3KO0 118217596 EC50 > 50000 nM T82702 C95ERM 118217608 EC50 > 50000 nM T82702 CM2U4C 118217609 EC50 > 22800 nM T82702 C9V0ZM 118217611 EC50 > 50000 nM T82702 CZ5L3N 118217612 EC50 > 50000 nM T82702 CCK3J9 118217851 EC50 > 50000 nM T82702 CO5I3V 118217852 EC50 > 17000 nM T82702 CD5TJ3 118217853 EC50 = 10600 nM T82702 C6HSC3 118217854 EC50 > 50000 nM T82702 CEKH57 118217858 EC50 > 50000 nM T82702 C7U0XR 118217863 EC50 > 50000 nM T82702 CDP0H5 118217865 EC50 > 50000 nM T82702 C82YDU 118217866 EC50 > 33000 nM T82702 CQ60HK 118217867 EC50 > 50000 nM T82702 C9N7VY 118217868 EC50 > 50000 nM T82702 C6LC7H 118217869 EC50 > 50000 nM T82702 CV9G4S 118217870 EC50 > 14000 nM T82702 C8PR3G 118217871 EC50 > 50000 nM T82702 CK85HV 118217875 EC50 > 50000 nM T82702 CT0DV4 118217911 EC50 > 50000 nM T82702 C1QPW5 118217915 EC50 = 7200 nM T82702 C3YTM2 118217920 EC50 > 50000 nM T82702 CU0T7K 118217922 EC50 = 5200 nM T82702 C0ETA2 118217925 EC50 > 50000 nM T82702 C89EDG 118217927 EC50 > 50000 nM T82702 C81QMJ 118217932 EC50 > 46100 nM T82702 C6X4IN 118217935 EC50 > 50000 nM T82702 CTNS59 118220706 EC50 = 48 nM T82702 CHY3F8 118220811 EC50 = 920 nM T82702 CD01CA 118526849 EC50 > 10000 nM T82702 CL8QZ9 118709251 EC50 = 1800 nM T82702 C3AE6V 118709252 EC50 = 700 nM T82702 C1T2CF 118709253 EC50 = 800 nM T82702 CDQV28 118709254 EC50 = 600 nM T82702 CV21FA 118709255 EC50 = 10000 nM T82702 CGS20Q 118709257 EC50 = 1500 nM T82702 C1N3VB 118709258 EC50 = 900 nM T82702 CMX6S5 118709259 EC50 = 50000 nM T82702 CC79WV 118709260 EC50 = 8800 nM T82702 CP3C1F 118714001 EC50 > 50000 nM T82702 C79CKF 118714035 EC50 > 25000 nM T82702 CFB78G 118714036 EC50 = 7800 nM T82702 CM5F8Z 118714037 EC50 > 25000 nM T82702 C2KET6 118714038 EC50 = 25000 nM T82702 CBZ75K 118724654 EC50 > 10000 nM T82702 CU4CW1 121313969 IC50 > 30000 nM T82702 CNGQ19 122179477 EC50 > 30000 nM T82702 C5L1AS 122184114 EC50 > 10000 nM T82702 CL7EY2 122184139 EC50 = 5400 nM T82702 CE87BY 122184140 EC50 = 400 nM T82702 C14FGL 122187534 EC50 > 50000 nM T82702 CRY8N5 122190169 EC50 = 4800 nM T82702 CTI2V5 122192293 EC50 > 50000 nM T82702 CI31MU 122194845 IC50 = 27400 nM T82702 COX7E3 122510453 EC50 > 24000 nM T82702 C4F9ZK 122669103 IC50 > 40000 nM T82702 CZH39M 122669106 IC50 > 40000 nM T82702 C0T8FO 122669173 IC50 > 40000 nM T82702 CD6X5P 122669265 EC50 > 50000 nM T82702 C0S7UB 122678562 IC50 > 40000 nM T82702 CY8S1P 122678563 IC50 > 40000 nM T82702 C0MUW2 122678576 IC50 > 40000 nM T82702 C2SQ9M 122678748 IC50 > 40000 nM T82702 CH1J6K 122678779 IC50 > 40000 nM T82702 CD9HN3 122678983 IC50 > 40000 nM T82702 CF39TE 122679031 IC50 > 40000 nM T82702 C0XWI7 127029952 EC50 = 630 nM T82702 CI3X9L 127049803 EC50 = 860 nM T82702 C2O5LX 127049804 EC50 > 3500 nM T82702 C8JW1U 129167185 EC50 = 25 nM T82702 C64QXT 130362615 EC50 = 290 nM T82702 CB62QX 131953519 EC50 = 144 nM T82702 CZ5H2B 132020452 IC50 > 50000 nM T82702 CP8A1Q 132020575 IC50 > 50000 nM T82702 C20HAT 134585236 EC50 = 11800 nM T82702 CTBR52 134585363 EC50 = 630 nM T82702 CHA58W 134585452 EC50 = 400 nM T82702 C6W3VL 134585536 EC50 = 4100 nM T82702 CCK2L8 134585538 EC50 = 420 nM T82702 CSN25F 134585580 EC50 = 4800 nM T82702 C6Q4RO 134585678 EC50 = 250 nM T82702 C7PZU3 134585707 EC50 = 420 nM T82702 CRL3O8 134585831 EC50 = 9400 nM T82702 CV0Y1T 134585845 EC50 > 20000 nM T82702 CAH0S5 134585890 EC50 = 3100 nM T82702 CZ2T3D 134585975 EC50 = 2450 nM T82702 C4TZI9 134586372 EC50 = 1680 nM T82702 CZPH61 134598642 EC50 = 3000 nM T82702 C63ONQ 135435181 EC50 = 5300 nM T82702 C8QMX0 135449328 EC50 = 10000 nM T82702 CY4MV6 135566354 EC50 > 30000 nM T82702 CX3VU1 136000590 EC50 > 30000 nM T82702 CRPQ42 136069494 IC50 > 50000 nM T82702 C7W4GE 136088954 EC50 > 30000 nM T82702 CUSE76 136098620 EC50 = 2100 nM T82702 C9DQ0A 136098621 EC50 = 4100 nM T82702 CQJ20H 136118727 EC50 = 1900 nM T82702 C6YB3M 136138768 EC50 = 5500 nM T82702 C4OVP2 136416802 EC50 > 30000 nM T82702 C7ZCT8 136416815 EC50 > 30000 nM T82702 C1ARX6 137297350 EC50 > 30000 nM T82702 C6B5US 137628648 EC50 > 50000 nM T82702 CK23OX 137633970 EC50 >= 50000 nM T82702 C07NWX 137637546 EC50 = 16700 nM T82702 C7VS2B 137645486 EC50 = 8330 nM T82702 CDO80K 137653078 EC50 = 2780 nM T82702 CZ4W3T 137656391 IC50 > 30000 nM T82702 C5B8OK 142505421 EC50 = 5900 nM T82702 CHB93R 142505434 EC50 = 7300 nM T82702 CRV6K9 142505445 EC50 = 2000 nM T82702 CYR1K0 142505452 EC50 = 57000 nM T82702 C71NAW 142505463 EC50 = 1300 nM T82702 CZM2D7 145963820 EC50 = 16 nM T82702 CKL63D 145965344 EC50 = 228 nM T82702 C13SNC 145965495 EC50 = 270 nM T82702 C4TL7G 145965870 EC50 = 254 nM T82702 C4H9UY 145966156 EC50 = 20 nM T82702 C4P3DR 145967002 EC50 = 190 nM T82702 CN78XB 145967589 EC50 > 30000 nM T82702 CG2A0S 145968399 EC50 > 30000 nM T82702 CA12HV 145969294 EC50 = 18000 nM T82702 CG27VL 145969403 EC50 = 520 nM T82702 CZF83O 145970182 EC50 = 2000 nM T82702 CYT8M9 145971562 EC50 = 175 nM T82702 CV9OM2 145973260 EC50 > 60000 nM T82702 CC8HN9 145973516 EC50 = 250 nM T82702 C0X3EB 145974156 EC50 = 1830 nM T82702 C13TQJ 145974494 EC50 = 18 nM T82702 CAYQ72 145974767 EC50 = 55 nM T82702 C60CDE 145975835 EC50 = 2860 nM T82702 CA3XR1 145976113 EC50 = 380 nM T82702 CE2O1P 145977892 EC50 = 36 nM T82702 C8G4QR 145982788 EC50 = 3200 nM T82702 CEX29U 145982851 EC50 = 4200 nM T82702 CU0V8B 145984255 EC50 = 14000 nM T82702 C2F8ZP 145984553 EC50 = 1400 nM T82702 CS4IU9 145984845 EC50 = 2400 nM T82702 CYRX35 145985210 EC50 = 1900 nM T82702 CP9Q8O 145985306 EC50 = 6500 nM T82702 C5TV7X 145985498 EC50 = 3400 nM T82702 CC89OI 148034311 IC50 > 40000 nM T82702 CE6V8Z 155511797 IC50 > 40000 nM T82702 CB4U3G 155515299 EC50 = 17000 nM T82702 CVH0P8 155519454 EC50 > 50118.72 nM T82702 CIUS51 155520682 EC50 = 3200 nM T82702 C20RGW 155522153 EC50 = 1500 nM T82702 CU5Z8T 155522788 IC50 > 40000 nM T82702 C0ASK5 155524887 EC50 = 3600 nM T82702 CS45AE 155524909 EC50 = 3300 nM T82702 C1DT9M 155525669 IC50 > 40000 nM T82702 CZW45D 155525803 EC50 > 50118.72 nM T82702 CXS9T8 155526989 IC50 > 40000 nM T82702 C0V6TI 155530389 EC50 = 1200 nM T82702 CO9N5H 155530678 IC50 > 40000 nM T82702 CS81FE 155530960 EC50 = 3000 nM T82702 C6B0LI 155532407 EC50 = 1600 nM T82702 CB5WR1 155532690 EC50 = 3700 nM T82702 CIUA10 155537856 IC50 > 40000 nM T82702 CC8F4Q 155538175 EC50 = 8400 nM T82702 CLO98T 155539150 EC50 > 50000 nM T82702 COP7X8 155539171 IC50 > 10000 nM T82702 C5T9KE 155542416 EC50 > 30000 nM T82702 C0V6EY 155543172 IC50 > 40000 nM T82702 CX7L0S 155544387 IC50 > 40000 nM T82702 CSK20E 155544524 IC50 > 40000 nM T82702 CTEC81 155544796 EC50 > 50000 nM T82702 C0N4JX 155552369 EC50 = 3500 nM T82702 C3WT2Q 155556441 EC50 > 30000 nM T82702 CBK1E5 155556708 IC50 > 40000 nM T82702 C3FI7U 155560819 IC50 > 40000 nM T82702 C5XH7Y 155560935 EC50 = 1500 nM T82702 C3Z6EL 155562317 EC50 > 20000 nM T82702 CC5FE7 155564581 EC50 > 30000 nM T82702 CA91EM 155564933 IC50 > 40000 nM T82702 CPF42S 155565257 IC50 > 40000 nM T82702 C9OC1G 155566505 EC50 = 1100 nM T82702 CUT84A 155568798 EC50 > 50000 nM T82702 C6KMU5 122184108 EC50 > 10000 nM T82702 CV5CO0 122184112 EC50 = 800 nM T82702 C63QAO 122184113 EC50 > 10000 nM T82702 CT3WD4 122184116 EC50 = 500 nM T82702 CBHT23 122184117 EC50 > 10000 nM T82702 CH1EJ7 122184118 EC50 = 1300 nM T82702 C13QFC 122184133 EC50 = 500 nM T82702 CO82BL 122184137 EC50 = 8800 nM T82702 CPM90L 122184138 EC50 = 900 nM T82702 D00DLU 16049480 EC50 = 250 nM T82702 D01BXE 9600409 EC50 = 990 nM T82702 D02DML 5281707 IC50 = 12000 nM T82702 D02TPY 25025860 IC50 = 3500 nM T82702 D02UID 16734800 IC50 = 1770 nM T82702 D04JSE 46200989 EC50 > 30000 nM T82702 D04KWH 176157 EC50 = 4950 nM T82702 D04SEX 446849 EC50 = 8600 nM T82702 D06HOI 44249821 EC50 > 25000 nM T82702 D09VTJ 441298 Ki = 27 nM T82702 D0B5FC 447912 EC50 = 8 nM T82702 D0BU8W 44219611 EC50 > 25000 nM T82702 D0C5SV 5280934 EC50 = 2 nM T82702 D0DQ2G 16043 EC50 = 2000 nM T82702 D0MU4A 5268 EC50 = 20000 nM T82702 D0PL4F 447905 Ki = 2000 nM T82702 D0Q0YS 644280 EC50 = 12600 nM T82702 D0T9VC 56840673 EC50 = 677 nM T82702 D0V0YM 24871527 EC50 = 5000 nM T82702 D0V4RZ 25113722 IC50 = 2160 nM T82702 D0V5SQ 68186 EC50 = 31600 nM T40556 D08HVE 679 IC50 = 280000000 nM T40556 D0E3SH 6918837 IC50 = 5 nM T40556 D0E7PQ 5311 IC50 = 10 nM T40556 D0L7LC 5352062 IC50 = 36 nM T40556 D00BYM 10461508 IC50 = 1070 nM T40556 D01LVE 57389999 IC50 = 39 nM T40556 D02YNI 9936746 Ki = 5.7 nM T40556 D03NJY 66577114 IC50 = 5300 nM T40556 D05ICT 132010322 Ki = 1.6 nM T40556 D06QBV 90647162 IC50 = 8 nM T40556 D07OFM 46943432 Ki = 23 nM T40556 D0G8BM 16722836 IC50 = 290 nM T40556 D0M2TS 71600087 IC50 = 1 nM T40556 D0O0LQ 11364421 IC50 = 25 nM T40556 D0PH9I 118693659 Ki = 5 nM T40556 D0XT6W 6918638 IC50 = 27 nM T40556 D0ZW4W 46907787 Ki = 5.3 nM T40556 D09FVR 122553422 IC50 < 11 nM T40556 D0HB3F 118340554 Ki < 1 nM T40556 D0KG9M 19910 IC50 = 980 nM T40556 D0SG9F 86566737 IC50 = 10 nM T40556 D09SFV 3973 IC50 = 12400 nM T40556 D0D3PX 46926350 IC50 = 19000 nM T40556 CL80QG 11820 IC50 = 73000 nM T40556 CZI4N9 13387 IC50 = 2660000 nM T40556 C5XSG3 19868 IC50 = 220000 nM T40556 C2BW3V 97075 IC50 = 34200 nM T40556 C4ZJO2 108402 IC50 = 6880000 nM T40556 CX0Z2S 205810 IC50 > 10000 nM T40556 CVG54O 209396 IC50 > 10000 nM T40556 CZX1K3 223771 IC50 > 200000 nM T40556 CD8OI6 251290 IC50 = 125892.54 nM T40556 C2IJU0 440987 IC50 = 39810.72 nM T40556 CJ6X2Y 572983 IC50 = 80000 nM T40556 CS7Z2U 584972 IC50 = 2870 nM T40556 CAT79Z 589098 IC50 > 100000 nM T40556 CPUC56 594190 IC50 = 101 nM T40556 CG5O0H 638578 IC50 = 18400 nM T40556 CG8C3X 651118 IC50 = 13300 nM T40556 C3CO8M 699832 IC50 = 210 nM T40556 CB3M7R 701320 IC50 = 47280 nM T40556 CB7ZY9 714750 IC50 = 5770 nM T40556 C4QD1V 723220 IC50 > 10000 nM T40556 CM1EX8 735746 IC50 = 3700000 nM T40556 COP70H 735747 IC50 = 260000 nM T40556 C4HEN5 739455 IC50 = 1000 nM T40556 CT41GY 747882 IC50 > 30000 nM T40556 CLN68U 750666 IC50 = 11000 nM T40556 CRN2X9 781532 IC50 = 47280 nM T40556 CX5U7E 781533 IC50 = 1910 nM T40556 CM71KW 786866 IC50 = 3000 nM T40556 CLC4D8 827656 IC50 > 10000 nM T40556 CT2J6Y 845994 IC50 = 27520 nM T40556 CB1Q6P 872951 IC50 = 71000 nM T40556 CV6DC3 878890 IC50 = 337 nM T40556 CS9GR8 893324 IC50 = 23060 nM T40556 CR65HV 975948 IC50 = 18720 nM T40556 C29JXM 984803 IC50 = 3020 nM T40556 C3UW5D 986642 IC50 > 10000 nM T40556 CQEF34 1002773 IC50 > 100000 nM T40556 CZ60SO 1015929 IC50 = 5730 nM T40556 CT48GV 1069056 IC50 = 530 nM T40556 C50QOJ 1069081 IC50 = 2280 nM T40556 CBG2A0 1078352 IC50 > 20000 nM T40556 CZP8B2 1090309 IC50 = 4800 nM T40556 CFA3Q8 1090310 IC50 = 4800 nM T40556 CV2ES8 1192817 IC50 = 130 nM T40556 CD0S4T 1220046 IC50 = 50750 nM T40556 C5TSY1 1244585 IC50 = 15530 nM T40556 CHP0C9 1380882 IC50 = 18000 nM T40556 CF3XV1 1382046 IC50 = 20000 nM T40556 C0TSA6 1395662 IC50 = 237.4 nM T40556 C92EYR 1503595 IC50 = 30000 nM T40556 CRT85V 1511056 IC50 = 69230 nM T40556 C2M0SE 1511198 IC50 = 1995.26 nM T40556 CJK1F0 1511199 IC50 = 1258.93 nM T40556 CZG1R8 1523399 IC50 = 3240 nM T40556 CI7UJ2 1523400 IC50 = 3740 nM T40556 C0A2LP 1523407 IC50 = 9680 nM T40556 C83WZI 1523409 IC50 = 4700 nM T40556 CY42VE 1534872 IC50 = 1530 nM T40556 CF1GQ2 1535153 IC50 = 1000 nM T40556 C7XRT1 1581020 IC50 = 1550 nM T40556 CCNQ31 1585889 IC50 = 1110 nM T40556 CP1L8I 1652717 IC50 = 1040 nM T40556 C31ITR 1895574 IC50 = 2100 nM T40556 CUVQ31 1922908 IC50 = 6600 nM T40556 CCJL62 2317823 IC50 > 10000 nM T40556 CP5GB0 2347699 IC50 = 769.2 nM T40556 C4T2JC 2371015 IC50 = 8940 nM T40556 C4Q0LV 2673048 IC50 > 100000 nM T40556 COZK67 2728636 IC50 = 43000 nM T40556 CDRT80 2782959 IC50 = 80900 nM T40556 CH95GA 2787707 IC50 = 8500 nM T40556 CHOL56 2824992 IC50 = 7500 nM T40556 C9V8HM 2841849 IC50 = 2100 nM T40556 C0EN8Y 2854307 IC50 > 10000 nM T40556 C8MB5Z 2874948 IC50 = 10980 nM T40556 C2OHC6 2927305 IC50 = 23000 nM T40556 C3DT1H 2973846 IC50 = 42230 nM T40556 CV9W7S 2988057 IC50 = 15800 nM T40556 C9PS6J 3109203 IC50 > 10000 nM T40556 CA89QB 3113698 IC50 = 370 nM T40556 C9RJG0 3132761 IC50 = 5360 nM T40556 CXD3U8 3152392 IC50 > 200000 nM T40556 CCS0Y2 3156673 IC50 = 738 nM T40556 CT1RG9 3293096 IC50 = 32230 nM T40556 C8GXW4 3319300 IC50 > 100000 nM T40556 CM1AE9 3370466 IC50 > 50118.72 nM T40556 CIE1C5 3499770 IC50 = 3400 nM T40556 CGE54P 3573716 IC50 > 50118.72 nM T40556 CS9M8A 3577407 IC50 > 50118.72 nM T40556 CJ4U6Y 3589423 IC50 = 5011.87 nM T40556 C2U9DI 3657707 IC50 = 39810.72 nM T40556 CPN2V4 3673391 IC50 > 50118.72 nM T40556 CYOV56 3681703 IC50 = 12589.25 nM T40556 C1KHJ6 3692581 IC50 = 3090 nM T40556 CB2ZP4 3721448 IC50 = 10940 nM T40556 C2P6IC 3846558 IC50 = 39000 nM T40556 C6KDA4 3900479 IC50 = 2103 nM T40556 CMDG67 3964313 IC50 = 50920 nM T40556 C42AQR 4102773 IC50 > 14000 nM T40556 C28EBX 4790771 IC50 = 39810.72 nM T40556 CY71BJ 4800411 Ki = 350 nM T40556 CR3SF5 4907545 IC50 = 5011.87 nM T40556 CWG19Q 4908238 IC50 = 19952.62 nM T40556 CB1HV6 4912924 IC50 > 100000 nM T40556 CXBG75 5125956 IC50 > 501187.23 nM T40556 C8BZ9Y 5325760 IC50 = 65000 nM T40556 CT8G2Z 6458480 IC50 > 50118.72 nM T40556 CEAN08 6611008 IC50 = 300 nM T40556 CLVK27 7731152 IC50 > 30000 nM T40556 C81TXG 8781434 IC50 = 2010 nM T40556 C5K3IF 9404764 IC50 = 34500 nM T40556 CC7IO0 9497211 IC50 = 890 nM T40556 C93EDN 10442296 IC50 > 100000 nM T40556 C5Y1WP 11128828 IC50 = 7000 nM T40556 C0BW3Q 11260691 IC50 = 84 nM T40556 CMJ01U 11283298 IC50 = 109 nM T40556 C6ALO2 11511524 Ki = 60 nM T40556 CE5K4J 11577250 IC50 = 25 nM T40556 CT53WA 12206142 IC50 > 200000 nM T40556 C1C6KY 12478742 Ki = 12000 nM T40556 C4H9EO 12488974 Ki = 21000 nM T40556 C34GWI 12622087 IC50 = 60000 nM T40556 CIG94A 13953713 IC50 = 19952.62 nM T40556 CTB86M 14774292 IC50 = 51000 nM T40556 CWPN42 15052068 IC50 = 12710 nM T40556 CQS67F 15944463 IC50 = 1090 nM T40556 CI82RX 15944465 IC50 > 30000 nM T40556 CP3EN5 15944506 IC50 = 1960 nM T40556 CP85DF 15944510 IC50 = 6490 nM T40556 CO8J4E 15944522 IC50 = 8220 nM T40556 C4E0UM 15944523 IC50 = 440 nM T40556 CTLV13 15944527 IC50 = 310 nM T40556 CN08ZF 15944528 IC50 = 9570 nM T40556 C1KAE2 15978962 IC50 = 33.9 nM T40556 CO3IL6 15990226 IC50 > 50118.72 nM T40556 CZ91JF 15990296 IC50 > 50118.72 nM T40556 C9K1AY 16228516 IC50 = 670 nM T40556 CCF3G5 16232084 IC50 > 50000 nM T40556 C1W7TE 16258532 IC50 = 10000 nM T40556 CP60ON 16258758 Ki = 1200 nM T40556 CE3X0C 16265714 Ki = 370 nM T40556 C25EUG 16272810 IC50 > 50118.72 nM T40556 CK2ES3 16313990 IC50 > 50118.72 nM T40556 CZ59FR 16316459 IC50 > 50118.72 nM T40556 CEN83U 16323492 IC50 > 50118.72 nM T40556 CM1R8O 16344932 IC50 = 31622.78 nM T40556 CQ3A6K 16371566 IC50 = 7400 nM T40556 CO6HM1 16480179 IC50 = 26000 nM T40556 CC17UZ 16654419 IC50 = 21270 nM T40556 CT5N9A 16654554 IC50 = 13850 nM T40556 CNK13T 16654568 IC50 = 11180 nM T40556 C4TC3X 16722832 IC50 = 130 nM T40556 CKJB19 16728035 IC50 = 18610 nM T40556 CY10PK 16728036 IC50 = 1640 nM T40556 CGFA68 16822024 Ki = 300 nM T40556 CO8M7K 17405877 IC50 = 199526.23 nM T40556 CIN8H3 17443248 IC50 = 19530 nM T40556 C9IP3Q 17446910 IC50 > 50118.72 nM T40556 CM09CN 17481591 IC50 = 24000 nM T40556 CLQ34F 17488246 IC50 = 160030 nM T40556 CO6KM2 17498966 IC50 > 100000 nM T40556 CVGU58 18536615 IC50 = 2900 nM T40556 CI8Z3Q 18536630 IC50 = 2500 nM T40556 C6Y4GF 18536633 IC50 = 3700 nM T40556 CDS15V 18536647 IC50 = 24000 nM T40556 C0DWP2 19596259 IC50 = 1810 nM T40556 CP7M5X 19704956 IC50 = 100 nM T40556 C4I2NX 20946734 IC50 > 50118.72 nM T40556 CDF52J 21680034 IC50 = 30000 nM T40556 C9IZ8A 21914263 IC50 = 4110000 nM T40556 C12TZA 22432992 IC50 > 50118.72 nM T40556 CXL15A 22433053 IC50 > 50118.72 nM T40556 CU9A5T 22696534 IC50 > 30000 nM T40556 C51GQD 24043179 Ki = 160000 nM T40556 CW5HI1 24156462 IC50 = 820 nM T40556 CLP9S1 24687782 IC50 > 50118.72 nM T40556 CIBE92 24789797 IC50 > 50118.72 nM T40556 COB70I 24789844 IC50 > 50118.72 nM T40556 C2JIY3 24790912 IC50 > 50118.72 nM T40556 C4S6OT 24906340 IC50 > 30000 nM T40556 CX2Q9M 24906350 IC50 = 6930 nM T40556 C49GBY 27604952 IC50 = 74000 nM T40556 CZ0JV1 27770210 IC50 = 6400 nM T40556 CN0J2C 29180108 IC50 > 50118.72 nM T40556 CAE73B 30342829 IC50 = 8180 nM T40556 C9OMZ0 30342838 IC50 = 3650 nM T40556 CQBK46 30342991 IC50 = 2050 nM T40556 CV6PQ8 30342999 IC50 = 810 nM T40556 CMQX14 30343069 IC50 = 4560 nM T40556 CI4AQ1 39129690 IC50 = 42000 nM T40556 C3UFS6 39791103 IC50 = 4800 nM T40556 C1OEL5 40889550 IC50 = 5200 nM T40556 CMN7L1 43286729 IC50 = 24000 nM T40556 C7KG1R 43286787 IC50 > 100000 nM T40556 C2P0IW 44243549 IC50 = 24600 nM T40556 C1C3QM 44269241 IC50 > 250000 nM T40556 C3VRO9 44557921 IC50 > 10000 nM T40556 C0GIA6 45103903 IC50 > 10000 nM T40556 CK3NP1 46249107 IC50 > 50118.72 nM T40556 C5HXW9 46249116 IC50 > 50118.72 nM T40556 CD06LA 46249215 IC50 = 10000 nM T40556 CCE1S0 47026724 IC50 = 27000 nM T40556 C3EL4J 47083668 IC50 = 8810 nM T40556 CT48OH 47108307 IC50 > 10000 nM T40556 C5FMU9 49169334 IC50 = 60000 nM T40556 C8H4PR 49766616 IC50 = 39040 nM T40556 CR87KB 49805721 Ki = 199.53 nM T40556 CN67BI 49805848 Ki = 398.11 nM T40556 C98BLM 49871817 IC50 = 26 nM T40556 C60BPW 49871818 IC50 > 10000000 nM T40556 CXC9K3 51003468 IC50 = 398.11 nM T40556 CI50XM 51063711 IC50 = 1700 nM T40556 C35MQH 51371083 IC50 > 20000 nM T40556 CTFL63 52100397 IC50 = 42230 nM T40556 CPSE59 52106219 IC50 = 10980 nM T40556 CWQ5G6 52106229 IC50 = 21130 nM T40556 CN5XV2 52106240 IC50 = 5210 nM T40556 C1PBE9 52233794 IC50 = 4630 nM T40556 C24YBT 52233800 IC50 = 11870 nM T40556 CHD35F 52233804 IC50 = 3340 nM T40556 CE4XV7 52233933 IC50 = 6540 nM T40556 CG3PR6 52912222 IC50 = 0.3981 nM T40556 CI68XL 52912223 IC50 = 280 nM T40556 CBXV52 52932793 IC50 = 251.19 nM T40556 CJE59U 52932930 IC50 = 1584.89 nM T40556 CSZ2T6 52932933 IC50 = 3162.28 nM T40556 CN87IR 52933159 IC50 = 794.33 nM T40556 CG6OL4 52933160 IC50 = 501.19 nM T40556 CP8Y9K 52933161 IC50 = 1258.93 nM T40556 CK8Z4P 52933165 IC50 = 3981.07 nM T40556 CKC17F 52933403 IC50 = 1258.93 nM T40556 CD08ZX 52933405 IC50 = 1000 nM T40556 C1T7VQ 52933407 IC50 = 1584.89 nM T40556 CE65VO 52933414 IC50 = 501.19 nM T40556 CFS84O 52933416 IC50 = 501.19 nM T40556 CO8VX9 52933655 IC50 = 1258.93 nM T40556 C6G7BE 52933893 IC50 = 794.33 nM T40556 C7VN1E 52934039 IC50 = 1000 nM T40556 CUZE18 52934122 IC50 = 501.19 nM T40556 CN16FE 52934128 IC50 = 6309.57 nM T40556 CTS13B 52934275 IC50 = 3981.07 nM T40556 CX3BI9 52934358 IC50 = 1995.26 nM T40556 CNOH36 52935183 IC50 = 251.19 nM T40556 CLRH53 52935478 IC50 = 1258.93 nM T40556 C53EFC 52935914 IC50 = 398.11 nM T40556 CXP76N 52936135 IC50 = 251.19 nM T40556 CJIB35 53054190 IC50 = 6000 nM T40556 C6V8YR 53054191 IC50 = 16000 nM T40556 C09HTR 53054200 IC50 = 1200 nM T40556 CUS8F7 53054236 IC50 = 7600 nM T40556 CX5QN4 53054237 IC50 = 20000 nM T40556 CD2TY9 53054238 IC50 = 11000 nM T40556 C47GAW 53054240 IC50 = 8200 nM T40556 CVH2G1 53054241 IC50 = 5600 nM T40556 CF9E2V 53054248 IC50 = 2600 nM T40556 CRWK92 53054249 IC50 = 5600 nM T40556 CSXI51 53054250 IC50 = 2000 nM T40556 CM12EL 53054251 IC50 = 3300 nM T40556 CY5L3J 53054252 IC50 = 4500 nM T40556 CWV76Y 53054258 IC50 = 1100 nM T40556 CIU8P7 53054259 IC50 = 500 nM T40556 CVX3R0 53054274 IC50 = 3300 nM T40556 CB05OM 53054276 IC50 = 1800 nM T40556 CLR97U 53054289 IC50 = 1000 nM T40556 CJ6E2Q 53054291 IC50 = 4400 nM T40556 C1WSZ4 53054297 IC50 = 2400 nM T40556 C7A2XC 53054319 IC50 = 3000 nM T40556 C0J1EO 53054320 IC50 = 6600 nM T40556 CK68UF 53054321 IC50 = 1200 nM T40556 CJY5S2 53054322 IC50 = 4200 nM T40556 C1YW5L 53054324 IC50 = 2800 nM T40556 C8Q6WG 53054325 IC50 = 1800 nM T40556 CJHR65 53268658 IC50 > 10000 nM T40556 CH6I4T 53268667 IC50 > 10000 nM T40556 CRG95D 53268718 IC50 = 1020 nM T40556 CQEF28 53308655 IC50 = 51200 nM T40556 C9V5LX 53318989 IC50 = 15.5 nM T40556 C7WVX3 54695746 IC50 = 2830 nM T40556 CEK3X6 54757749 IC50 = 23200 nM T40556 C1D3WH 54757750 IC50 = 9700 nM T40556 C1DZ7Y 54757751 IC50 = 7700 nM T40556 C6W5OZ 54757752 IC50 = 7500 nM T40556 C1KWY4 54759170 IC50 = 10000 nM T40556 CM8Y7O 56697168 IC50 = 13260 nM T40556 C7HK2C 56924692 IC50 = 2600 nM T40556 CTVM34 56929801 IC50 = 380.19 nM T40556 CX6SD9 56950289 IC50 = 3200 nM T40556 CZ6NE0 56950420 IC50 = 2500 nM T40556 CJ5BE9 56950421 IC50 = 5200 nM T40556 CL96VQ 56950422 IC50 = 3000 nM T40556 CCLD98 56950423 IC50 = 13000 nM T40556 CZD7G2 56950424 IC50 = 6500 nM T40556 CPQ0B7 56950425 IC50 = 7400 nM T40556 CL90DK 56950426 IC50 = 1000 nM T40556 CF9IJ1 56950561 IC50 = 1300 nM T40556 CH24QC 56950562 IC50 = 12000 nM T40556 CU62NO 56950563 IC50 = 17000 nM T40556 CRD86M 56950564 IC50 = 15000 nM T40556 CNQ2L5 56950565 IC50 = 22000 nM T40556 CB3A1Z 56950566 IC50 = 10000 nM T40556 C5ADP4 56950567 IC50 = 17000 nM T40556 CFW0D1 57339435 IC50 = 1258.93 nM T40556 C56SWR 57344430 IC50 = 6200 nM T40556 C3ZXF4 57344431 IC50 = 36 nM T40556 CU74JQ 57344432 IC50 = 1100 nM T40556 CEK82U 57344527 IC50 = 2200 nM T40556 CE71PA 57344528 IC50 = 86 nM T40556 C6OZU2 57344531 IC50 = 200 nM T40556 CE37LA 57344606 IC50 = 190 nM T40556 CEP6Q1 57345408 IC50 < 500 nM T40556 CCU1P9 57388845 IC50 = 5700 nM T40556 C0Z9HP 57389114 IC50 = 2100 nM T40556 C31KUT 59149763 Ki = 251.19 nM T40556 CF8B4E 60498769 IC50 = 5000 nM T40556 CYL1B0 66553124 IC50 = 1900 nM T40556 CKC51O 66553125 IC50 = 4800 nM T40556 CW8K1P 67173666 IC50 = 7943.28 nM T40556 CPD6G3 67192581 IC50 = 1258.93 nM T40556 CX17NA 67195278 IC50 = 501.19 nM T40556 CPY59D 67195867 IC50 = 25118.86 nM T40556 C0QK5F 67814495 IC50 = 250 nM T40556 CN3KZ8 68161075 IC50 = 398.11 nM T40556 C49IOA 68161669 IC50 = 501.19 nM T40556 CJ7N3M 68184870 IC50 = 1258.93 nM T40556 CT4Z2A 68184871 IC50 = 501.19 nM T40556 CEX74I 68186034 IC50 = 5011.87 nM T40556 CCE3I0 68199877 IC50 = 33 nM T40556 C25INY 68204735 IC50 = 1258.93 nM T40556 C6KWC8 69236418 IC50 > 200000 nM T40556 CMC7V5 70664240 IC50 = 1258.93 nM T40556 CDY89S 70680609 IC50 > 50000 nM T40556 C1I6OH 70681167 IC50 = 7943.28 nM T40556 C7GJW9 70681170 IC50 = 630.96 nM T40556 C8H4JX 70681173 IC50 = 794.33 nM T40556 C6NYK2 70681174 IC50 = 501.19 nM T40556 C8KBJ0 70683271 IC50 = 1258.93 nM T40556 CXD3F9 70691699 IC50 = 398.11 nM T40556 C9L0KD 70699440 IC50 = 386 nM T40556 CV7OR2 70699441 IC50 = 380.19 nM T40556 C76BEK 71271375 IC50 = 390 nM T40556 C0HTY9 71271805 IC50 = 880 nM T40556 CJ90CI 71271897 IC50 = 220 nM T40556 C76ZPW 71271926 IC50 = 600 nM T40556 CR96WH 71271969 IC50 = 4400 nM T40556 C2P4GJ 71272064 IC50 = 360 nM T40556 C5YBX2 71272103 IC50 = 730 nM T40556 C7VJK4 71272293 IC50 = 180 nM T40556 C1UZ4Q 71272605 IC50 = 2300 nM T40556 CFSP50 71297183 IC50 = 790 nM T40556 COZ1E0 71297184 IC50 = 4100 nM T40556 CB2NY9 71297185 IC50 = 4100 nM T40556 CS1BL2 71450122 IC50 = 880 nM T40556 CL8Y9N 71450297 IC50 = 1258.93 nM T40556 CUY20J 71459124 IC50 = 470 nM T40556 C6CQT5 71462842 IC50 = 6309.57 nM T40556 CWUE65 71532084 IC50 = 27 nM T40556 CMJC68 71615940 Ki = 3.1 nM T40556 CONT42 71615943 Ki = 6.4 nM T40556 C6U5KC 71615944 Ki = 4.1 nM T40556 CTXM79 71616053 Ki = 1.5 nM T40556 C2U7NS 71616054 Ki = 2.9 nM T40556 CLZ7X1 71616055 Ki = 14 nM T40556 CXLN73 71616297 Ki = 48 nM T40556 C7UQH0 71616300 Ki = 2.4 nM T40556 C47LAI 71616301 Ki = 4.4 nM T40556 CR3M1X 71616302 Ki = 9.8 nM T40556 C93NFZ 71616418 Ki = 32 nM T40556 CN1H9P 71616658 Ki = 4.5 nM T40556 CY20JZ 71616659 Ki = 68 nM T40556 C25ZDV 71616989 Ki = 3.6 nM T40556 C82EAI 71617108 Ki = 9.4 nM T40556 C1UA6X 71617219 Ki = 5.8 nM T40556 C4O7ZL 71617338 Ki = 68 nM T40556 C1SHR7 71617458 Ki = 12 nM T40556 CYI2A3 71617461 Ki = 19 nM T40556 CE91KU 71617462 Ki = 3.7 nM T40556 C7BU8M 71621544 Ki = 6.3 nM T40556 C4MJ0T 71624784 IC50 = 640 nM T40556 CIX91F 71624785 IC50 = 1700 nM T40556 C1D8GF 71624786 IC50 = 1500 nM T40556 C3R9WA 71624787 IC50 = 3900 nM T40556 CLQ1X8 71624896 IC50 = 2600 nM T40556 COW9G4 71624897 IC50 = 544 nM T40556 CODK30 71624901 IC50 = 1360 nM T40556 CI15JC 71624902 IC50 = 1380 nM T40556 CLZ7C8 71624903 IC50 = 1170 nM T40556 CLA71B 71661332 IC50 = 3700 nM T40556 CW5F3S 71661333 IC50 = 10000 nM T40556 C7US6G 71661335 IC50 = 22800 nM T40556 CP0C3Q 71661522 IC50 = 23800 nM T40556 C13DUN 71661524 IC50 = 3300 nM T40556 C9WZO5 71661707 IC50 = 3500 nM T40556 C7FW1U 71661708 IC50 = 2600 nM T40556 CG3U8D 71661709 IC50 = 2400 nM T40556 CAYC45 71661710 IC50 = 2500 nM T40556 C0TK5C 71661712 IC50 = 230 nM T40556 C1FD9C 71661885 IC50 = 2200 nM T40556 C74UGA 71661886 IC50 = 570 nM T40556 C1VXA5 71664045 IC50 = 50700 nM T40556 CWJR48 71664046 IC50 = 2600 nM T40556 C7GY3D 71664047 IC50 = 4400 nM T40556 CX8B7F 71717163 IC50 = 58.7 nM T40556 CG10TU 71720056 IC50 = 180 nM T40556 CS26GP 71747837 IC50 > 10000 nM T40556 CIPN50 71760902 Ki = 15 nM T40556 C74CSP 71811952 EC50 = 7100 nM T40556 CMZU93 71811973 EC50 = 280 nM T40556 CZQ4G1 71812037 EC50 = 75 nM T40556 CHDB19 71812048 Ki = 210 nM T40556 CA1F7L 71812065 Ki = 91 nM T40556 C1IHP6 71812067 Ki = 250 nM T40556 CX73WV 71862498 IC50 = 63280 nM T40556 CD1FE6 71935082 IC50 = 1900 nM T40556 CIYP36 71938587 IC50 = 3000 nM T40556 CL0NM3 71942353 IC50 = 24000 nM T40556 C7FVU5 71970469 IC50 = 11720 nM T40556 C1OGC5 71975056 IC50 = 21000 nM T40556 CGP24T 72201024 IC50 = 2511.89 nM T40556 CA81BL 72201025 IC50 = 4100 nM T40556 CA71SN 72203613 IC50 = 14 nM T40556 C9M6QY 72547793 Ki = 2.6 nM T40556 CTQ9S3 72548029 Ki = 5.6 nM T40556 CUI57F 72548032 Ki = 17 nM T40556 CW4QJ6 72548735 Ki = 14 nM T40556 C4L6PB 72549215 Ki = 140 nM T40556 C01LXD 72549905 Ki = 58 nM T40556 C64NRP 72550116 Ki = 13 nM T40556 C4VBJ1 72684073 IC50 = 1258.93 nM T40556 C2AFW1 72702849 IC50 = 398.11 nM T40556 C3R1IL 72703043 IC50 = 100000 nM T40556 CK9O6W 72705811 IC50 = 6309.57 nM T40556 CIW9K7 72713634 IC50 = 66000 nM T40556 C3W5VQ 72713635 IC50 = 74000 nM T40556 CBS16L 72713636 IC50 = 28000 nM T40556 C1LUB0 72713637 IC50 = 42000 nM T40556 C1Q6MO 72945553 IC50 = 290 nM T40556 C97BCW 72945554 IC50 = 74 nM T40556 CEW3O7 72945555 IC50 = 250 nM T40556 CL7EB1 73347805 IC50 = 91 nM T40556 CBD0N5 73349345 IC50 = 72 nM T40556 CUG1T8 73350913 IC50 = 29 nM T40556 CEH74A 73350914 IC50 = 42 nM T40556 C2C0ZX 73352391 IC50 = 398.11 nM T40556 C9VQ7H 73352402 IC50 = 1500 nM T40556 CD9NK1 73353867 IC50 = 380 nM T40556 CJY67C 73355395 IC50 = 2500 nM T40556 C3LQ4W 73425805 IC50 = 20 nM T40556 C2WDM8 73891130 IC50 = 1 nM T40556 C6VDW2 75373087 IC50 = 107410 nM T40556 CQOV07 75375570 IC50 > 200000 nM T40556 CW5A7G 76070631 IC50 = 126 nM T40556 CFZ65N 76071650 IC50 = 8 nM T40556 C0FD7H 76071652 IC50 = 15 nM T40556 CC3OJ7 76072013 IC50 = 9 nM T40556 CS7U4H 76072259 IC50 = 5 nM T40556 CQ78NK 76310219 IC50 = 158.49 nM T40556 CM4J8Q 76317442 IC50 = 251.19 nM T40556 CIN36T 76318560 IC50 = 7000000 nM T40556 CM7TH3 76328466 IC50 = 5011.87 nM T40556 C0T5NK 76335637 IC50 = 1000 nM T40556 CW7BS4 76534645 IC50 = 18 nM T40556 C9NE5G 76683426 IC50 = 30 nM T40556 CW6MD3 76683643 IC50 = 80 nM T40556 C3NIR2 76902013 IC50 = 37 nM T40556 CLW3A6 76902201 IC50 = 49 nM T40556 C46HRP 76902203 IC50 = 190 nM T40556 CKT41J 77108173 IC50 = 20 nM T40556 C8FRL6 77108189 IC50 = 10 nM T40556 CU6O0X 77461280 IC50 < 50 nM T40556 C5TB9S 77843982 Ki = 34 nM T40556 CI87ZD 77844001 IC50 = 1 nM T40556 CS6XE0 77846025 Ki = 12.2 nM T40556 COZ8S1 78319129 Ki = 77 nM T40556 C2TG5M 78320028 IC50 = 10 nM T40556 CTGH72 78320336 IC50 = 10 nM T40556 C85MTQ 78320816 Ki = 180 nM T40556 CCW9M4 78320817 Ki = 12 nM T40556 CN54HC 78321130 IC50 = 1.8 nM T40556 CX78QI 78321451 Ki = 43 nM T40556 CJA4F5 78322398 Ki = 47.8 nM T40556 CDZK41 78322399 Ki = 201 nM T40556 CZP9K2 78322539 IC50 = 140 nM T40556 CR6B4F 78323579 IC50 = 30 nM T40556 C3G2YK 78323818 IC50 = 20 nM T40556 C6BE7U 78325043 IC50 = 78 nM T40556 C4IF8T 78425807 Ki = 0.62 nM T40556 CVF12D 78428091 IC50 = 14 nM T40556 C4X6VZ 82104609 IC50 = 780 nM T40556 C4LA6F 86208116 IC50 = 637 nM T40556 CQUO30 86270617 Ki = 450 nM T40556 C1YFW8 86270651 Ki = 7.1 nM T40556 CHKW02 86270831 Ki = 26 nM T40556 CHK64J 86270834 Ki = 0.87 nM T40556 CFE7R3 86270928 Ki = 0.73 nM T40556 CE1V5Z 86270929 Ki = 16 nM T40556 C5KG4I 86271129 IC50 = 3.7 nM T40556 CT6BG3 86271751 Ki = 84 nM T40556 C81AKZ 86271752 EC50 = 280 nM T40556 C5WKC6 86271987 IC50 = 8 nM T40556 CV3YT8 86273096 IC50 = 27 nM T40556 CWPU56 86273098 IC50 = 31 nM T40556 C3EN0I 86273586 IC50 = 34 nM T40556 CB9AL4 86287631 IC50 < 11 nM T40556 CS4QR8 86287687 Ki = 120 nM T40556 C7SNT4 86287688 Ki = 17 nM T40556 CI8BA9 86287690 Ki = 11 nM T40556 COA7X4 86287755 Ki = 5.5 nM T40556 CB8JP3 86287958 Ki = 11 nM T40556 CDG13U 86295201 Ki = 54 nM T40556 C5M8RB 86295909 IC50 < 200 nM T40556 C8ONF2 86296101 IC50 = 35 nM T40556 CFV1S8 86296389 IC50 < 14 nM T40556 CX0KF8 86299084 Ki = 38 nM T40556 CS9F7V 86299086 Ki = 450 nM T40556 C9XR0G 86299218 Ki = 270 nM T40556 CUE87M 86299220 Ki = 1600 nM T40556 C6RT3M 86299506 EC50 > 10000 nM T40556 CXFG10 86301666 Ki = 3.8 nM T40556 C9W1SR 86581390 Ki = 1.3 nM T40556 CRN51L 86581538 Ki = 0.6 nM T40556 CE7B1X 86582295 IC50 = 3 nM T40556 C7IPH4 86582916 Ki = 2.1 nM T40556 C53QEW 86669224 IC50 = 6309.57 nM T40556 C7ZDO0 86808440 IC50 = 33160 nM T40556 C0RD6L 87056019 IC50 = 20 nM T40556 CQC6V8 87397080 IC50 > 100000 nM T40556 CY7P2N 89656146 Ki = 13 nM T40556 CW7PG2 89656147 IC50 = 58 nM T40556 C4JXL8 89656405 Ki = 680 nM T40556 CMSH53 89657387 Ki = 38 nM T40556 CGE9F1 89657420 Ki = 32 nM T40556 CEDL57 89657555 EC50 = 2480 nM T40556 CRU32W 89657560 Ki = 1.3 nM T40556 C8FXA7 89657583 Ki = 1.2 nM T40556 C1FOK3 90016835 Ki = 7 nM T40556 CXD3A6 90017103 EC50 = 370 nM T40556 CV8R0Z 90017113 Ki = 230 nM T40556 CUR5Z8 90017358 Ki = 22 nM T40556 CCB43O 90018193 Ki = 5.1 nM T40556 CZ54IL 90019075 Ki = 5.5 nM T40556 C2XQD4 90019266 Ki = 16 nM T40556 C4YE1K 90019789 Ki = 71 nM T40556 C8GN5H 90019850 Ki = 110 nM T40556 CV41WZ 90019957 Ki = 1900 nM T40556 CHK91R 90020090 Ki = 9 nM T40556 CU6CZ1 90026274 Ki = 450 nM T40556 CO82NI 90026512 Ki = 1700 nM T40556 CN4MG2 90026969 Ki = 890 nM T40556 CHC5I8 90027770 Ki = 13 nM T40556 C0T5SJ 90028262 Ki = 120 nM T40556 C13BOQ 90032394 Ki = 1700 nM T40556 CLQN32 90104652 IC50 = 10100 nM T40556 C68NDT 90364429 IC50 = 77 nM T40556 CPOG43 90387291 Ki = 41 nM T40556 CP25VC 90387467 Ki = 194 nM T40556 CZJ8W9 90387575 Ki = 16.1 nM T40556 C3JXP5 90387666 Ki = 98.1 nM T40556 C1EJ7F 90387844 IC50 = 200 nM T40556 CSW41E 90387917 Ki = 478 nM T40556 CW4IF5 90388035 Ki = 116 nM T40556 CED71H 90388046 Ki = 2182 nM T40556 C37YQH 90388075 Ki = 1948 nM T40556 C3C7GD 90388178 Ki = 1500 nM T40556 C6O2BH 90388309 Ki = 80 nM T40556 C1HD8T 90388367 Ki = 867 nM T40556 CFAE47 90388486 Ki = 98.8 nM T40556 C01MOG 90388523 Ki = 8322 nM T40556 CICK10 90388552 Ki = 824 nM T40556 CX90PZ 90395609 Ki = 19.7 nM T40556 C0UEK8 90395610 Ki = 18.5 nM T40556 CEYR46 90395611 Ki = 41.2 nM T40556 C5WG4S 90395612 Ki = 335 nM T40556 CHK85V 90395617 Ki < 0.5 nM T40556 CME05X 90395619 Ki < 0.5 nM T40556 C3WS5V 90395622 Ki = 30.6 nM T40556 C2D0LZ 90395625 Ki = 1.1 nM T40556 CNZ1V4 90395627 Ki = 7 nM T40556 CS4P9H 90395630 Ki = 44.3 nM T40556 CD94HJ 90395631 Ki = 2.8 nM T40556 CV75CK 90395632 IC50 > 1000 nM T40556 C62DJX 90395643 Ki = 22.5 nM T40556 C5XRI2 90395644 Ki = 4.2 nM T40556 CMX16I 90395646 Ki = 2.7 nM T40556 CQB83M 90395649 Ki = 2.8 nM T40556 CVK1M3 90395718 Ki = 52.3 nM T40556 CI28DM 90395720 Ki = 3.8 nM T40556 CW94AZ 90395721 Ki = 3.1 nM T40556 CYMD60 90395722 Ki = 42.6 nM T40556 C8UC4Z 90395724 Ki = 4.2 nM T40556 C1PJX2 90395725 Ki = 26.9 nM T40556 C49IVE 90395727 Ki = 139 nM T40556 C1KPZ5 90395734 Ki = 1.6 nM T40556 CFQ92A 90395738 Ki = 58.2 nM T40556 CR70LI 90395752 Ki = 1.4 nM T40556 C20LRN 90413429 Ki = 420 nM T40556 CLMV91 90413480 EC50 = 280 nM T40556 C3LC7M 90415492 Ki = 280 nM T40556 CD1Q4I 90417643 Ki = 17 nM T40556 CCF4T3 90466145 IC50 < 200 nM T40556 C1I7QN 90654869 IC50 > 30000 nM T40556 C1A6EO 90654871 IC50 = 7550 nM T40556 CCAL04 90654872 IC50 = 3180 nM T40556 C8F4IL 90667393 IC50 = 1995.26 nM T40556 CC76KI 90667394 IC50 = 1584.89 nM T40556 C07UWH 90667395 IC50 = 63095.73 nM T40556 CI79XN 90667396 IC50 = 19952.62 nM T40556 CYQ91J 90667397 IC50 = 6309.57 nM T40556 C4WCZ6 90667398 IC50 = 31622.78 nM T40556 C1J9HN 90667399 IC50 = 19952.62 nM T40556 C3WIR5 90667400 IC50 = 6309.57 nM T40556 CX1A3E 90667401 IC50 = 6309.57 nM T40556 C6FA3S 90667402 IC50 = 6309.57 nM T40556 CBS30L 90667403 IC50 = 3981.07 nM T40556 CV6DO1 90667404 IC50 = 630.96 nM T40556 C95ZKF 90667405 IC50 = 1258.93 nM T40556 CZP13T 90667406 IC50 = 794.33 nM T40556 CIA7N6 90667407 IC50 = 1000 nM T40556 CEA70Y 90667408 IC50 = 1584.89 nM T40556 C40KGW 90667409 IC50 = 794.33 nM T40556 CPMJ06 90667410 IC50 = 794.33 nM T40556 C64QIN 90667411 IC50 = 630.96 nM T40556 C83ORG 90667412 IC50 = 12589.25 nM T40556 C03DRI 90667413 IC50 = 1000 nM T40556 C16WGN 90667414 IC50 = 3981.07 nM T40556 CO92PS 90667415 IC50 = 10000 nM T40556 CLV2G0 90667416 IC50 = 1258.93 nM T40556 CJQZ54 90667417 IC50 = 630.96 nM T40556 CDRA20 90667418 IC50 = 1995.26 nM T40556 C0RX4B 90667452 IC50 = 50 nM T40556 C8HL5V 90667453 IC50 = 290 nM T40556 C3IE7F 90667454 IC50 = 360 nM T40556 C37GOB 90667455 IC50 = 100 nM T40556 C3PFG1 90670355 IC50 = 1690 nM T40556 C08KZL 90670356 IC50 = 15100 nM T40556 CD3P8Y 91215896 IC50 = 16000 nM T40556 CZ39RM 91668224 IC50 < 300 nM T40556 CYF7O2 91668539 IC50 = 50.12 nM T40556 C2JXG5 91668540 IC50 = 2511.89 nM T40556 CZ0H2Y 91668542 IC50 = 19952.62 nM T40556 C1BOU8 91758311 IC50 = 9 nM T40556 CB7Q8G 91809474 IC50 = 1400 nM T40556 CD7P5Y 91809475 IC50 = 250 nM T40556 CJ35EM 91809476 IC50 = 60 nM T40556 C8WX4I 91810827 IC50 < 5 nM T40556 CHOS65 91820723 IC50 = 25118.86 nM T40556 C0TNJ7 91820724 IC50 = 3981.07 nM T40556 C0N1GO 91826363 IC50 = 15 nM T40556 C8XL0I 91826394 IC50 < 11 nM T40556 CAZ9M0 91826677 IC50 = 3981.07 nM T40556 CEN52P 91826678 IC50 = 6309.57 nM T40556 CD0W7N 91971372 IC50 = 350 nM T40556 CY1WR2 92019884 IC50 = 2120000 nM T40556 C9WB3G 95828281 IC50 = 60000 nM T40556 CJ4MO9 95991007 IC50 > 100000 nM T40556 C3BIT0 100922929 IC50 = 90000 nM T40556 CU62EH 101481444 Ki = 25000 nM T40556 CB19IE 102358573 IC50 = 13000 nM T40556 CU91GC 105539824 IC50 = 26000 nM T40556 COD1I8 105539836 IC50 = 2580 nM T40556 C3M4CS 105539837 IC50 = 450 nM T40556 C3L5KU 105539840 IC50 = 450 nM T40556 C15PLR 105539841 IC50 = 2290 nM T40556 C9L7AG 105539842 IC50 = 730 nM T40556 CMDU18 105539860 IC50 = 410 nM T40556 C1W3XP 112499930 IC50 = 1900 nM T40556 CYX7T2 117072549 IC50 > 100000 nM T40556 C6EKA2 117689397 IC50 = 79 nM T40556 C4L1MR 117689434 IC50 = 107 nM T40556 CM9H5G 117689436 IC50 = 76 nM T40556 CUA1Z2 117689648 IC50 = 148 nM T40556 C8C6GE 117772437 Ki = 1.1 nM T40556 C5RF3K 117775483 Ki = 1.7 nM T40556 C24ZCQ 117775856 Ki = 0.6 nM T40556 C1RSV4 117833983 IC50 > 100000 nM T40556 C3PIB1 117833991 IC50 = 11800 nM T40556 CXL1W7 117834061 IC50 = 807 nM T40556 CG0LW1 117834596 IC50 = 968 nM T40556 C4OYH6 117834599 IC50 > 100000 nM T40556 C2QDF9 117834602 IC50 = 2890 nM T40556 CHF9V8 117834605 IC50 = 2760 nM T40556 C6B0TG 117834606 IC50 = 904 nM T40556 C0TLH3 117834615 IC50 = 474 nM T40556 CNJ58G 117834616 IC50 = 11000 nM T40556 CXK54D 117834619 IC50 = 3890 nM T40556 CN15HA 117834638 IC50 = 31500 nM T40556 CA0RF9 117834640 IC50 = 1660 nM T40556 C4K3JM 117834641 IC50 = 18800 nM T40556 CP8NJ4 117834648 IC50 = 4530 nM T40556 CE2TK1 117841251 IC50 = 13000 nM T40556 C0WZL6 117841252 IC50 = 12900 nM T40556 CH0L6O 117841253 IC50 = 51900 nM T40556 CD6H0A 117841254 IC50 = 13000 nM T40556 CVM0I2 117841255 IC50 = 562 nM T40556 C2JD5A 117841259 IC50 = 1170 nM T40556 CXVE97 117841261 IC50 = 479 nM T40556 C7PS8I 117841263 IC50 = 2050 nM T40556 CCU4G9 117841264 IC50 = 3170 nM T40556 CHS4W1 117841265 IC50 = 11900 nM T40556 CAK0P3 117841267 IC50 = 1620 nM T40556 C8YK5G 117841268 IC50 = 20700 nM T40556 CH6MJ5 117841269 IC50 = 2860 nM T40556 CP8KY3 117841270 IC50 = 860 nM T40556 C1NFO3 117891931 IC50 = 12 nM T40556 C4O8MX 117928476 IC50 < 1000 nM T40556 CV9T2S 118021357 IC50 = 420 nM T40556 C20BJO 118021398 IC50 = 920 nM T40556 CF1V6O 118021399 IC50 = 410 nM T40556 CA82SI 118021476 IC50 = 15 nM T40556 C9TJD6 118021554 IC50 = 9500 nM T40556 C7V1TN 118021622 IC50 = 2990 nM T40556 C3GM0W 118021678 IC50 = 24 nM T40556 C3BR8O 118021718 IC50 = 2 nM T40556 CDCF34 118021720 IC50 = 50 nM T40556 CSW7D8 118021721 IC50 = 510 nM T40556 C3LAW9 118021764 IC50 = 710 nM T40556 C4SCT5 118021773 IC50 = 460 nM T40556 C1IY8X 118021799 IC50 = 150 nM T40556 CD1P6E 118021813 IC50 = 2890 nM T40556 CGPK87 118021821 IC50 = 25 nM T40556 C72DWE 118021851 IC50 = 270 nM T40556 CA5CO3 118021879 IC50 = 160 nM T40556 CCR09V 118021930 IC50 = 368 nM T40556 CEG49X 118021977 IC50 = 750 nM T40556 C4JE7G 118021984 IC50 = 150 nM T40556 CF9YQ2 118022046 IC50 = 13000 nM T40556 CXAC70 118022070 IC50 = 240 nM T40556 C48NXS 118022125 IC50 = 49 nM T40556 C2MSO5 118022126 IC50 = 20000 nM T40556 C80GPR 118022184 IC50 = 250 nM T40556 C57CSH 118022209 IC50 = 240 nM T40556 C06EWP 118022266 IC50 = 1600 nM T40556 C7M9BE 118022285 IC50 = 11500 nM T40556 C97LFH 118022380 IC50 = 5 nM T40556 C8EGS1 118022691 IC50 = 3 nM T40556 C0MU6N 118022972 IC50 = 910 nM T40556 CUL98O 118060057 IC50 < 1000 nM T40556 CR15YL 118078883 IC50 = 370 nM T40556 CHDQ27 118078887 IC50 = 380 nM T40556 CN73AQ 118078912 IC50 = 43000 nM T40556 C6ZD3F 118078985 IC50 = 1600 nM T40556 CW6D8E 118079032 IC50 = 1400 nM T40556 C68LAH 118079235 IC50 = 60 nM T40556 CQJ6E2 118079293 IC50 < 100 nM T40556 C8S3BF 118079489 IC50 = 380 nM T40556 C9D8FA 118079501 IC50 = 100 nM T40556 CHP05V 118079652 IC50 = 420 nM T40556 CWN5B3 118079664 IC50 > 50000 nM T40556 C6VF5A 118079690 IC50 = 1600 nM T40556 CQ03GL 118079722 IC50 > 25000 nM T40556 CQ0BM1 118079985 IC50 > 50000 nM T40556 CIE48C 118080085 IC50 = 760 nM T40556 CU74JC 118080153 IC50 = 1700 nM T40556 CS1N3M 118080263 IC50 = 14000 nM T40556 C7D8OM 118080305 IC50 = 790 nM T40556 C6IJZ3 118080562 IC50 = 260 nM T40556 CMU0G5 118093990 IC50 = 1218 nM T40556 C61SNT 118094033 IC50 = 342 nM T40556 C0QT8P 118094069 IC50 = 596 nM T40556 C3G1DO 118116651 IC50 = 2.3 nM T40556 CLJ43Y 118117152 IC50 = 11 nM T40556 C6A1RW 118120978 IC50 = 10120 nM T40556 CHB87O 118120979 IC50 = 2890 nM T40556 CQ5V6F 118121011 IC50 = 4960 nM T40556 C5RS9G 118137754 Ki = 8.9 nM T40556 CZH8X7 118137759 Ki = 1.5 nM T40556 CYA1M0 118137762 IC50 = 2 nM T40556 CBGI40 118137765 Ki = 11 nM T40556 C29BNE 118137780 Ki = 1.9 nM T40556 CAB1X0 118137789 Ki = 1.5 nM T40556 CH9Z3Y 118137820 Ki = 2.8 nM T40556 C8A0CL 118137846 Ki = 3.4 nM T40556 CT8J9Y 118137861 Ki = 7.3 nM T40556 C8P3YF 118137879 Ki = 100 nM T40556 CGQY32 118137892 Ki = 3.8 nM T40556 CR0H9F 118137913 Ki = 2 nM T40556 CM06ZO 118138005 Ki = 0.8 nM T40556 C5Q4MC 118138006 IC50 = 1.3 nM T40556 C5P9RD 118169070 IC50 < 150 nM T40556 CAD1B6 118196369 IC50 < 5 nM T40556 CK50FQ 118196502 IC50 < 5 nM T40556 CPTF61 118200167 IC50 = 13900 nM T40556 CJ8YA2 118200170 IC50 = 5900 nM T40556 CZAI75 118200236 IC50 = 1940 nM T40556 C4Y5DB 118237331 IC50 = 63 nM T40556 C4P7MG 118277818 Ki = 27 nM T40556 CZ7D5J 118288035 IC50 = 150 nM T40556 CKG9S0 118288047 Ki = 99 nM T40556 C8ZQL1 118288049 Ki = 470 nM T40556 CGR63N 118288050 IC50 = 100 nM T40556 C73MQC 118317783 IC50 = 650 nM T40556 C5VQM0 118340530 Ki = 21.5 nM T40556 CG7WB4 118340538 Ki = 0.5 nM T40556 C13IJX 118340548 Ki = 2.6 nM T40556 C90KHI 118340551 Ki = 2 nM T40556 CS1D3I 118340553 Ki = 387 nM T40556 C6T9PS 118340596 Ki = 16.7 nM T40556 CQD5U2 118340603 Ki = 0.7 nM T40556 CR26LY 118340612 Ki < 1 nM T40556 CX09DZ 118340631 IC50 > 1000 nM T40556 C25VBU 118340646 Ki = 78 nM T40556 CI6E9H 118340650 Ki = 3.4 nM T40556 CZN8G5 118340653 Ki = 66.5 nM T40556 CFH02N 118340663 Ki < 1 nM T40556 C5T2HE 118340668 Ki = 2.4 nM T40556 CZT5M4 118340676 Ki = 6.3 nM T40556 C3RM5Q 118340684 Ki < 1 nM T40556 COR5G3 118340697 Ki = 1.7 nM T40556 C0GJZ5 118340710 Ki = 15.8 nM T40556 CF2C0W 118340714 Ki = 77.9 nM T40556 CM5TN1 118340720 Ki < 1 nM T40556 CXVK68 118340726 Ki = 3.1 nM T40556 CM34GO 118340729 Ki < 1 nM T40556 CPI9J0 118340741 Ki = 31 nM T40556 CS8KG3 118340760 Ki = 0.8 nM T40556 C35BHR 118340789 Ki = 28.4 nM T40556 C7IAX1 118340796 Ki = 1.2 nM T40556 C1MHG0 118340829 Ki = 1 nM T40556 CN1K0V 118340834 Ki = 4.9 nM T40556 C60DGX 118340843 Ki < 1 nM T40556 CE58WP 118509530 IC50 = 1.3 nM T40556 CXT73W 118509541 IC50 = 5 nM T40556 C8ZLN9 118693661 IC50 = 1.7 nM T40556 CR0PO8 118693673 Ki = 1.585 nM T40556 C8YNI5 118693928 Ki = 3.981 nM T40556 CPN74M 118719856 IC50 = 794.33 nM T40556 CE8DL3 118719857 IC50 = 630.96 nM T40556 COEU47 118719858 IC50 = 1000 nM T40556 CX05SW 118719859 IC50 = 630.96 nM T40556 CRCG07 118719860 IC50 = 501.19 nM T40556 C03XDG 118719861 IC50 = 501.19 nM T40556 C3ML2F 118719862 IC50 = 794.33 nM T40556 CZ67WF 118719863 IC50 = 25118.86 nM T40556 C0HR9Y 118719864 IC50 = 630.96 nM T40556 C7F4EP 118719865 IC50 = 316.23 nM T40556 CA40QV 118719866 IC50 = 630.96 nM T40556 CZ8QI6 118719867 IC50 = 794.33 nM T40556 C8NRI9 118719868 IC50 = 1000 nM T40556 C3Y2WT 118719869 IC50 = 1000 nM T40556 C52HPM 118719870 IC50 = 501.19 nM T40556 CUT97H 118719871 IC50 = 630.96 nM T40556 CBE68N 118719872 IC50 = 1000 nM T40556 C29WRE 118719873 IC50 = 794.33 nM T40556 C8J0TY 118719874 IC50 = 1000 nM T40556 CZR10C 118719875 IC50 = 3981.07 nM T40556 C35AWU 118719876 IC50 = 2511.89 nM T40556 C4OFG7 118721302 IC50 = 16300 nM T40556 CA8HW2 118721303 IC50 > 100000 nM T40556 CZY31K 118721304 IC50 > 50118.72 nM T40556 CYGS87 118721305 IC50 = 1584.89 nM T40556 C9O0IC 118721631 IC50 = 69900 nM T40556 CE9Y5W 118721632 IC50 = 7860 nM T40556 C63SEK 118727389 IC50 = 17900 nM T40556 C8NWB4 118727390 IC50 = 7800 nM T40556 C7F9XN 118727392 IC50 = 7200 nM T40556 C90BQI 118727394 IC50 = 78600 nM T40556 C9YJN5 118727397 IC50 = 63000 nM T40556 C8LA9O 118727400 IC50 = 29700 nM T40556 C6YUB8 118727401 IC50 = 20000 nM T40556 CGL92E 118727402 IC50 = 5600 nM T40556 CA82PM 118727403 IC50 = 427 nM T40556 CI4CQ2 118732060 IC50 = 2260 nM T40556 CIGL03 118732061 IC50 = 2060 nM T40556 C4ZA8M 118732062 IC50 > 10000 nM T40556 CQ71XK 118732063 IC50 = 8330 nM T40556 C8TRM7 118732064 IC50 = 7340 nM T40556 C6Z5CE 118732065 IC50 > 10000 nM T40556 CEXW89 118732066 IC50 > 10000 nM T40556 CTDN06 118732067 IC50 = 9310 nM T40556 CR07PK 118732068 IC50 = 5820 nM T40556 CJG89V 118732069 IC50 = 220 nM T40556 CDV60F 118732070 IC50 = 760 nM T40556 CFVW10 118732071 IC50 = 500 nM T40556 CAFB70 118732072 IC50 = 120 nM T40556 CN6D1A 118732073 IC50 = 400 nM T40556 CV3U7I 118732074 IC50 = 800 nM T40556 CM5YS0 118732075 IC50 = 300 nM T40556 CJWX45 118732076 IC50 = 60 nM T40556 CX35ZI 118732077 IC50 = 460 nM T40556 CQ84KV 118732078 IC50 = 140 nM T40556 CF57ZY 118732079 IC50 = 220 nM T40556 CL6U1T 118732080 IC50 = 170 nM T40556 C0XIA1 118732081 IC50 = 930 nM T40556 C7V9JG 118732082 IC50 = 100 nM T40556 CS2V9Y 118732083 IC50 = 790 nM T40556 CA3S1C 118732084 IC50 = 250 nM T40556 CU95AV 118740117 IC50 > 84000 nM T40556 C87ZPY 118796358 IC50 > 100000 nM T40556 CRF4G8 118796361 IC50 = 1121 nM T40556 CWS6Y5 118796362 IC50 = 3681 nM T40556 C9VQX4 118863284 IC50 = 0.7 nM T40556 C38TSJ 118863314 IC50 = 4.6 nM T40556 CQ2GC8 118863432 Ki = 7.3 nM T40556 CE4PK9 118863469 Ki = 4.1 nM T40556 CF9J8E 118918705 IC50 = 1700 nM T40556 CA3Z8O 118918714 IC50 = 2800 nM T40556 C8GLJ3 118918720 IC50 = 7200 nM T40556 C2ZY3U 118932975 IC50 > 10000 nM T40556 CC14FI 118933132 IC50 = 4500 nM T40556 CGO91Y 118933136 IC50 = 17000 nM T40556 CFMJ96 119081417 IC50 = 2900 nM T40556 C8AZ4C 119081691 IC50 = 2500 nM T40556 CUWX94 119081692 IC50 = 65 nM T40556 C9MQF0 119098887 IC50 = 30652 nM T40556 C0QX4D 119098889 IC50 = 23576 nM T40556 CBD7I6 121232405 IC50 = 19952.62 nM T40556 C4JN5Q 121237855 IC50 = 2400 nM T40556 C4AU0X 121237856 IC50 > 120000 nM T40556 C7A2UY 121237857 IC50 = 1500 nM T40556 CBN53Q 121271705 IC50 = 8500 nM T40556 CGBI67 121271742 IC50 = 13000 nM T40556 CPU76D 121271756 IC50 > 20000 nM T40556 CN4X9G 121271781 IC50 = 8900 nM T40556 CB83MK 121271792 IC50 = 11000 nM T40556 C0F6MH 121277645 IC50 > 200000 nM T40556 C0FA3C 121277864 IC50 = 16000 nM T40556 CP1NH2 121277975 IC50 = 4500 nM T40556 C0XVY8 121277987 IC50 = 8000 nM T40556 CHO97R 121277993 IC50 = 12000 nM T40556 COW87E 121278062 IC50 = 7000 nM T40556 C1PGY8 121278155 IC50 > 20000 nM T40556 C3GD2W 121335190 IC50 = 460 nM T40556 C81OYL 121335218 IC50 > 20000 nM T40556 C83RUE 121335260 IC50 = 8200 nM T40556 CECP26 121335281 IC50 = 1500 nM T40556 C1HR3M 121335283 IC50 > 20000 nM T40556 C2EP5S 121335312 IC50 = 2300 nM T40556 CNW25A 121338193 IC50 = 6100 nM T40556 C5JYP8 121338332 IC50 > 20000 nM T40556 C5ML2V 121338401 IC50 > 20000 nM T40556 C3JMB8 121338437 IC50 > 20000 nM T40556 CF25LT 121338490 IC50 > 20000 nM T40556 C5US9K 121338530 IC50 = 19200 nM T40556 CMF5D4 121338574 IC50 = 17200 nM T40556 C0VF7X 121338589 IC50 > 20000 nM T40556 CQ30XW 121342392 IC50 = 3600 nM T40556 CNM34X 121342393 IC50 = 3400 nM T40556 CXI0K8 121342398 IC50 = 600 nM T40556 C9O4RD 121342404 IC50 = 1200 nM T40556 CJMF61 121342523 IC50 = 1800 nM T40556 CQKU78 121342528 IC50 = 7900 nM T40556 C8CV7M 121365342 IC50 > 20000 nM T40556 C41LZU 121365398 IC50 = 18000 nM T40556 CNJ4A0 121365442 IC50 = 8500 nM T40556 C12KNG 121365488 IC50 = 3700 nM T40556 C8YE5F 121365519 IC50 = 3100 nM T40556 C46MHD 121372830 IC50 = 4200 nM T40556 CIW10X 121372875 IC50 = 7300 nM T40556 CFH51D 121372877 IC50 = 5600 nM T40556 C7W2KQ 121372879 IC50 = 13000 nM T40556 C7P2EW 121372880 IC50 > 20000 nM T40556 CDC61P 121372884 IC50 = 5900 nM T40556 C34YHN 121372887 IC50 = 13000 nM T40556 C6EID7 121372897 IC50 > 20000 nM T40556 C94PWO 121372898 IC50 = 4600 nM T40556 CL67ME 121372914 IC50 = 7300 nM T40556 CQ8ZL9 121372939 IC50 = 20000 nM T40556 C3I8SV 121372947 IC50 = 9600 nM T40556 CKYL73 121372990 IC50 = 4200 nM T40556 CQ0AL8 121372997 IC50 = 4000 nM T40556 C32SNH 121373004 IC50 = 870 nM T40556 C4UD7J 121373027 IC50 = 6400 nM T40556 CV9KF4 121373031 IC50 > 20000 nM T40556 CE2VJ4 121373032 IC50 = 9200 nM T40556 CZ30EX 121373033 IC50 = 12000 nM T40556 C1HRP7 121373036 IC50 > 20000 nM T40556 CP0OX4 121373042 IC50 = 15000 nM T40556 CDQV23 121373043 IC50 = 13000 nM T40556 CVO7B2 121373072 IC50 = 2200 nM T40556 CD9PJ2 121373074 IC50 = 3900 nM T40556 C57ZDO 121373154 IC50 = 4600 nM T40556 CS9XW0 121373155 IC50 = 8600 nM T40556 CYDN26 121373156 IC50 = 3700 nM T40556 CI84KM 121373164 IC50 = 3800 nM T40556 CK03TO 121373206 IC50 = 16000 nM T40556 C4G2QK 121373220 IC50 > 20000 nM T40556 C57GXL 121373316 IC50 = 4100 nM T40556 C04UKS 121373365 IC50 = 5400 nM T40556 CDH8M4 121373418 IC50 = 4200 nM T40556 C1TK3U 121373476 IC50 > 20000 nM T40556 CW1HV7 121373599 IC50 = 11000 nM T40556 C2V6AX 121373769 IC50 = 9500 nM T40556 C47QXT 121376807 IC50 = 13000 nM T40556 C9XWC0 121376818 IC50 = 12000 nM T40556 C0QKG5 121376850 IC50 = 4800 nM T40556 CP6R5B 121382912 IC50 = 4000 nM T40556 C51UXY 121414852 IC50 = 160 nM T40556 C19VLJ 121414853 IC50 = 130 nM T40556 CL5SB9 121414854 IC50 = 15 nM T40556 CWC98G 121499171 IC50 = 25118.86 nM T40556 C6E0UL 122164589 Ki = 12.59 nM T40556 C5PKZ6 122164734 IC50 = 70 nM T40556 C67WYM 122164963 Ki = 7.943 nM T40556 CEF87B 122164964 Ki > 1000 nM T40556 CO9J5W 122179607 IC50 = 1258.93 nM T40556 C3WOE8 122179608 IC50 = 6309.57 nM T40556 CW03JY 122179609 IC50 = 1000 nM T40556 CHNS18 122179610 IC50 = 3162.28 nM T40556 C2Q0OY 122179611 IC50 = 1258.93 nM T40556 C9GPL4 122179612 IC50 = 6309.57 nM T40556 CZX41C 122179613 IC50 = 3981.07 nM T40556 CJDK15 122179614 IC50 = 7943.28 nM T40556 CSF76G 122179615 IC50 = 1995.26 nM T40556 CY7U0Z 122179616 IC50 = 794.33 nM T40556 C1MV9L 122179617 IC50 = 1258.93 nM T40556 CJ81BV 122179618 IC50 = 15848.93 nM T40556 CZ69QO 122180530 IC50 > 50118.72 nM T40556 C7D5VP 122180531 IC50 = 39810.72 nM T40556 CRY84E 122180532 IC50 = 5011.87 nM T40556 C0J1AY 122180533 IC50 = 50118.72 nM T40556 CPIV02 122180534 IC50 > 50118.72 nM T40556 CC9XH7 122180535 IC50 > 50118.72 nM T40556 C0IWE1 122180536 IC50 > 501187.23 nM T40556 CEF19P 122180537 IC50 = 10000 nM T40556 C20LOD 122180538 IC50 = 19952.62 nM T40556 C73OMU 122180539 IC50 = 6309.57 nM T40556 CZSB51 122180540 IC50 = 6309.57 nM T40556 CJ4LO2 122180541 IC50 = 15848.93 nM T40556 C4TB0F 122180542 IC50 = 10000 nM T40556 CTXL15 122180543 IC50 = 39810.72 nM T40556 CUDY80 122180544 IC50 = 12589.25 nM T40556 C0SC2Y 122180545 IC50 = 25118.86 nM T40556 CR6T4G 122180546 IC50 = 25118.86 nM T40556 CHJG86 122180547 IC50 = 158489.32 nM T40556 CYZV97 122180548 IC50 = 15848.93 nM T40556 C0AIU8 122180549 IC50 = 12589.25 nM T40556 CPUS31 122180550 IC50 = 12589.25 nM T40556 CD62RB 122180551 IC50 = 6309.57 nM T40556 C8UCV9 122180552 IC50 = 3162.28 nM T40556 C72NLB 122180553 IC50 = 5011.87 nM T40556 CR0K5P 122180554 IC50 = 7943.28 nM T40556 CZ6L2N 122180555 IC50 = 3981.07 nM T40556 CKH49I 122180556 IC50 = 3162.28 nM T40556 CS4PD6 122180557 IC50 = 794.33 nM T40556 CWC9I4 122180558 IC50 = 1000 nM T40556 CE7SL5 122180559 IC50 = 630.96 nM T40556 CR6YD4 122180560 IC50 = 125.89 nM T40556 C8HCK6 122180561 IC50 = 1995.26 nM T40556 CX9C6Y 122180562 IC50 = 794.33 nM T40556 CPZ67Y 122180563 IC50 = 3162.28 nM T40556 CN1LE0 122180564 IC50 = 5011.87 nM T40556 C4ITM8 122180892 IC50 = 13000 nM T40556 CFCA87 122180893 IC50 = 13000 nM T40556 CZRJ29 122180894 IC50 = 13000 nM T40556 C8RE2M 122180895 IC50 = 14000 nM T40556 C54NBV 122180896 IC50 = 16000 nM T40556 C26RAL 122180897 IC50 = 18000 nM T40556 CC35RW 122180898 IC50 = 25000 nM T40556 C7E3VM 122180899 IC50 = 25000 nM T40556 C2UQW0 122180900 IC50 = 34000 nM T40556 C67LPS 122180901 IC50 = 40000 nM T40556 C3FC0Z 122180902 IC50 = 44000 nM T40556 CSR48T 122180903 IC50 = 46000 nM T40556 CVI96R 122180904 IC50 > 50000 nM T40556 CZB15E 122180905 IC50 = 9000 nM T40556 C6V0UQ 122180906 IC50 = 13000 nM T40556 COR80H 122180907 IC50 = 25000 nM T40556 CFVN54 122180908 IC50 = 29000 nM T40556 CXP8T3 122180909 IC50 = 44000 nM T40556 CE29NL 122180910 IC50 = 47000 nM T40556 CR78FH 122180911 IC50 = 49000 nM T40556 CB1M0U 122180912 IC50 > 50000 nM T40556 CGLF82 122181547 IC50 = 6309.57 nM T40556 CZGK74 122181548 IC50 = 10000 nM T40556 C9P3GX 122181549 IC50 = 10000 nM T40556 C3QJ5L 122181550 IC50 = 15848.93 nM T40556 C3NC4V 122181552 IC50 = 7943.28 nM T40556 C41ZXJ 122181555 IC50 = 1584.89 nM T40556 C6I3VJ 122181557 IC50 = 630.96 nM T40556 C7CJR2 122181559 IC50 = 12589.25 nM T40556 CP5Z1C 122181560 IC50 = 15848.93 nM T40556 C61RTG 122181561 IC50 = 12589.25 nM T40556 CT62FG 122181571 IC50 = 10000 nM T40556 CJ8B1U 122187515 Ki = 7950 nM T40556 CHI14C 122187516 Ki = 4500 nM T40556 CUX72G 122187517 Ki > 10000 nM T40556 CI86PH 122187518 Ki > 10000 nM T40556 CD24VL 122187519 Ki = 1400 nM T40556 C8ZLB5 122187520 Ki > 10000 nM T40556 C6OGU0 122187521 Ki = 970 nM T40556 CW84YE 122187522 Ki = 8.7 nM T40556 CH83IY 122187523 Ki = 37 nM T40556 C6CWM2 122187524 Ki = 46 nM T40556 C24AKR 122187525 Ki = 29 nM T40556 CZ3E7H 122187526 Ki = 100 nM T40556 CO25IW 122191031 IC50 >= 10000 nM T40556 C4WGV6 122191040 IC50 = 4000 nM T40556 CDY43J 122191048 IC50 >= 10000 nM T40556 C79NTO 122446081 IC50 = 14 nM T40556 C0LNZ9 122446098 IC50 = 21 nM T40556 C5EQJ0 122467457 IC50 = 4290 nM T40556 C4ME9H 122467464 IC50 > 30000 nM T40556 C56NAS 122467465 IC50 = 4170 nM T40556 C35LXF 122467467 IC50 > 30000 nM T40556 CEJ5W3 122467468 IC50 = 3440 nM T40556 C80AFH 122467469 IC50 = 2550 nM T40556 C5BY0I 122467470 IC50 = 600 nM T40556 CO8R3Y 122467472 IC50 = 5640 nM T40556 C3E6UB 122467476 IC50 = 4840 nM T40556 CQ71FH 122467477 IC50 > 30000 nM T40556 C6V7LS 122467478 IC50 = 1210 nM T40556 C7QV4I 122467480 IC50 > 30000 nM T40556 C12RVQ 122467483 IC50 > 30000 nM T40556 CLAE37 122467484 IC50 = 1500 nM T40556 CY2CD5 122467486 IC50 = 510 nM T40556 CM4NH1 122467488 IC50 = 5290 nM T40556 COCT-54 122467494 IC50 > 30000 nM T40556 CKC3B1 122467495 IC50 = 4100 nM T40556 CNI3H2 122467498 IC50 = 1120 nM T40556 C62IDL 122470439 IC50 = 10 nM T40556 C7VJH3 122512239 IC50 = 12.59 nM T40556 C6DS2X 122553424 IC50 < 11 nM T40556 CU8L1O 122553479 IC50 = 12 nM T40556 CN51WG 122588588 IC50 < 0.5 nM T40556 C3C8QO 122588611 IC50 = 3 nM T40556 C0KE5N 122588642 IC50 = 2 nM T40556 CWJD15 122705990 IC50 > 10000 nM T40556 CIR48B 123146482 IC50 = 501.19 nM T40556 CR9T6N 123814574 IC50 = 1000 nM T40556 C7GWV1 124098192 IC50 = 18800 nM T40556 C5VQN1 124429951 IC50 = 3980 nM T40556 C20LTP 125383342 IC50 = 77 nM T40556 CR98TS 125994265 IC50 > 10000 nM T40556 C4GYP3 126521168 IC50 = 32 nM T40556 CL2PG5 126521180 IC50 = 18 nM T40556 CQV90I 126521354 IC50 = 28 nM T40556 C0HJV7 126521430 IC50 > 999 nM T40556 CN6FI1 126521537 IC50 = 2 nM T40556 C1DOG4 126521586 IC50 = 14 nM T40556 CRY0S6 126563516 IC50 = 12 nM T40556 CN0D6M 126563562 IC50 = 10 nM T40556 CKB36S 126563576 IC50 = 7 nM T40556 CX79NH 126563597 IC50 = 14 nM T40556 C2K5XG 126563611 IC50 = 17 nM T40556 CZ06NR 126563612 IC50 = 36 nM T40556 CM5P2Z 126563615 IC50 = 30 nM T40556 C15ILF 126564427 IC50 = 7 nM T40556 CROY39 126564463 IC50 = 7 nM T40556 CHO12Y 126564469 IC50 > 10000 nM T40556 CB2AS4 126564470 IC50 = 6 nM T40556 CBW08I 126564471 IC50 = 12 nM T40556 CD78GB 126564481 IC50 = 10 nM T40556 CU8CA9 126564486 IC50 = 6 nM T40556 CQW6P1 126564822 IC50 = 11 nM T40556 CQS5T2 126564831 IC50 = 23 nM T40556 CNP2L7 126564832 IC50 = 13 nM T40556 C58PNK 126564833 IC50 = 15 nM T40556 CHPV09 126564847 IC50 = 10 nM T40556 CJZW04 126564858 IC50 = 13 nM T40556 C4WXN8 126772498 IC50 = 24910 nM T40556 CM8EB4 126961333 IC50 = 16700 nM T40556 C0MR6T 126961716 Ki = 970 nM T40556 CJR0V7 127025419 IC50 = 1258.93 nM T40556 CZ93IW 127025420 IC50 = 398.11 nM T40556 C5FV9L 127025697 IC50 = 501.19 nM T40556 C8N5UA 127025979 IC50 = 2511.89 nM T40556 C7M2GL 127025980 IC50 = 15848.93 nM T40556 C2LYR4 127025981 IC50 = 12589.25 nM T40556 C8GLF2 127025982 IC50 = 199.53 nM T40556 CMG7C1 127026579 IC50 = 38900 nM T40556 C57IHP 127026582 IC50 > 50000 nM T40556 CF9QV5 127026591 IC50 > 50000 nM T40556 C4MY5E 127026593 IC50 > 50118.72 nM T40556 C7OQT2 127026594 IC50 = 1584.89 nM T40556 C62OFC 127026595 IC50 = 794.33 nM T40556 C0C1HZ 127028091 IC50 > 50000 nM T40556 COXV68 127029808 IC50 = 5560 nM T40556 CS37AQ 127030405 IC50 < 300 nM T40556 C0DF1I 127030450 IC50 > 30000 nM T40556 CV81XG 127030451 IC50 = 2980 nM T40556 CNG8Y1 127030726 IC50 = 85 nM T40556 C6B4HD 127030768 IC50 = 1580 nM T40556 C5XN8O 127030774 IC50 = 3510 nM T40556 C6FI7V 127031094 IC50 = 470 nM T40556 CB7X6C 127031095 IC50 = 3870 nM T40556 C7GQI0 127031954 IC50 = 1160 nM T40556 CEVK16 127032241 IC50 = 1670 nM T40556 CVOS94 127032857 IC50 = 3130 nM T40556 CH14FC 127032939 IC50 = 8100 nM T40556 CR2A7U 127033172 IC50 = 1190 nM T40556 C1SA9P 127033473 IC50 > 30000 nM T40556 C0P5EA 127033474 IC50 = 4270 nM T40556 CBT9C7 127033475 IC50 = 1170 nM T40556 C30AKN 127033476 IC50 = 460 nM T40556 CIG3Q9 127033567 IC50 = 20400 nM T40556 CS4NG8 127033568 IC50 = 26400 nM T40556 C0JYH2 127033770 IC50 = 210 nM T40556 CG20LF 127034058 IC50 = 4900 nM T40556 CCK36M 127034059 IC50 = 4810 nM T40556 C2JOB7 127034595 IC50 = 400 nM T40556 C3R6VW 127034596 IC50 = 620 nM T40556 CRH92V 127034597 IC50 = 1720 nM T40556 C7V0HE 127034598 IC50 = 120 nM T40556 CV07YO 127038801 IC50 <= 1000 nM T40556 C4RGQ7 127043287 IC50 > 50118.72 nM T40556 CF3Z9G 127043292 IC50 > 50118.72 nM T40556 CA3VI9 127043861 IC50 = 10000 nM T40556 CCSJ69 127043862 IC50 > 50118.72 nM T40556 CJT6N0 127043863 IC50 = 25118.86 nM T40556 CEG46M 127043864 IC50 = 7943.28 nM T40556 CL8S6X 127043872 IC50 > 50118.72 nM T40556 CEAN18 127043873 IC50 > 50118.72 nM T40556 CZP0D9 127043874 IC50 = 10000 nM T40556 C7Y1IB 127043875 IC50 = 12589.25 nM T40556 CH4BE8 127043876 IC50 > 50118.72 nM T40556 CWP65X 127043881 IC50 = 19952.62 nM T40556 CO62HW 127044040 IC50 = 39810.72 nM T40556 CE0CG1 127044041 IC50 > 50118.72 nM T40556 CJ7YT3 127044046 IC50 > 50118.72 nM T40556 CAN9K0 127044332 IC50 > 50118.72 nM T40556 CH1MJ8 127044333 IC50 > 50118.72 nM T40556 CP15DV 127044334 IC50 > 50118.72 nM T40556 CU7X9E 127044335 IC50 > 50118.72 nM T40556 CXN63Y 127044336 IC50 > 50118.72 nM T40556 CLN5S3 127044787 IC50 > 50118.72 nM T40556 CX4M3R 127044824 IC50 > 50118.72 nM T40556 CZ5H7K 127045294 IC50 = 10000 nM T40556 CQOL84 127045572 IC50 = 39810.72 nM T40556 CGA71L 127048256 IC50 = 61917 nM T40556 CH6T5J 127048257 IC50 = 67479 nM T40556 C60SZQ 127048258 IC50 = 47095 nM T40556 C6BT3U 127048317 IC50 > 20000 nM T40556 C9DY4Z 127048318 IC50 = 8000 nM T40556 C5AV7U 127049278 IC50 = 31421 nM T40556 C50BMV 127049279 IC50 = 5861 nM T40556 CTFY41 127049280 IC50 = 32430 nM T40556 CVE71A 127049281 IC50 = 19165 nM T40556 C73TND 127049282 IC50 = 3778 nM T40556 CEN16G 127049286 IC50 = 44000 nM T40556 C9C0MB 127049631 IC50 = 3500 nM T40556 C8MXQ7 127049932 IC50 > 20000 nM T40556 C2VC3L 127050405 IC50 = 1147 nM T40556 CWFM08 127050492 IC50 = 81300 nM T40556 CTF4N2 127051087 IC50 > 100000 nM T40556 CD2T1E 127051228 IC50 = 780 nM T40556 CPS8R6 127051229 IC50 = 850 nM T40556 C12KXI 127051477 IC50 > 20000 nM T40556 CRZ3A6 127051526 IC50 = 670 nM T40556 CR0P6Q 127051527 IC50 = 3730 nM T40556 CLSZ47 127051725 IC50 = 23005 nM T40556 CMY93U 127051726 IC50 = 47359 nM T40556 CY8V1A 127051727 IC50 > 100000 nM T40556 CXZT48 127052023 IC50 > 100000 nM T40556 C9V3AX 127052165 IC50 = 1490 nM T40556 C2OHP4 127052166 IC50 = 1380 nM T40556 CS60GZ 127052167 IC50 = 1050 nM T40556 C2RB3T 127052469 IC50 = 2990 nM T40556 CHA05V 127052470 IC50 = 770 nM T40556 C5EYK2 127053005 IC50 > 20000 nM T40556 CG6AY7 127053006 IC50 > 20000 nM T40556 CGM6W4 128963618 IC50 > 20000 nM T40556 CT2M0R 129214093 Ki = 10.4 nM T40556 C7C0WK 129606900 IC50 = 79.43 nM T40556 CO8Z2N 129900111 IC50 = 34000 nM T40556 CTLO82 130345485 Ki = 70 nM T40556 CJ6VO1 130345500 Ki = 190 nM T40556 C4DJO5 130345531 Ki = 1500 nM T40556 CIJ23L 130345532 Ki = 13 nM T40556 CX32JZ 130345556 Ki = 3300 nM T40556 CO0L1R 130345558 Ki = 15 nM T40556 C9L1OG 130345579 Ki = 2.3 nM T40556 COI68Y 130345587 Ki = 2800 nM T40556 C8JV7L 130345597 Ki = 820 nM T40556 C0RTS8 130345606 Ki = 4.2 nM T40556 C98WYE 130345614 Ki = 33 nM T40556 C1XDL5 130345617 Ki = 2.1 nM T40556 C5FUX9 130357671 Ki = 250 nM T40556 CG2RM3 130357741 Ki = 2.7 nM T40556 C7NEB1 130471695 IC50 > 10800 nM T40556 CLA09E 130471696 IC50 > 20000 nM T40556 CWNY27 130471723 IC50 > 12100 nM T40556 CXW1B4 130471724 IC50 > 14500 nM T40556 C1EN7A 130471730 IC50 > 13900 nM T40556 C2HD6P 130471733 IC50 = 14500 nM T40556 C5DFI7 130471761 IC50 > 20000 nM T40556 CDLE96 130471765 IC50 > 20000 nM T40556 C1C8OB 130471770 IC50 > 9500 nM T40556 CDC32I 130471775 IC50 > 14250 nM T40556 C3D7HE 130471777 IC50 > 20000 nM T40556 CFI30C 130471784 IC50 > 11450 nM T40556 C7TJA6 130471785 IC50 > 15000 nM T40556 CDUX50 130471789 IC50 > 15000 nM T40556 C8VAM6 130471790 IC50 > 12950 nM T40556 CN80UV 130471849 IC50 > 20000 nM T40556 CEV5I3 130471855 IC50 > 15000 nM T40556 CE1K3M 130471876 IC50 > 11900 nM T40556 CFTG42 130472058 IC50 > 9950 nM T40556 C5P2ED 130472268 IC50 > 15000 nM T40556 C7B6CZ 130472269 IC50 = 15500 nM T40556 CED70X 130472274 IC50 > 10000 nM T40556 CNUG19 131740828 Ki = 1100 nM T40556 CK0B6N 131985884 IC50 = 1700 nM T40556 CUN18W 132005225 IC50 = 10800 nM T40556 CD84OI 132005228 IC50 = 6000 nM T40556 C7ASP9 132005246 IC50 = 18800 nM T40556 CE89ZR 132010072 Ki = 1.3 nM T40556 C0W9DE 132010081 Ki = 6.9 nM T40556 C39MLW 132010085 Ki = 1.2 nM T40556 CKB6N5 132010104 Ki = 1.1 nM T40556 CYE3D7 132010164 Ki = 1 nM T40556 C7WP0Z 132010280 Ki = 1.1 nM T40556 CFN06J 132010408 Ki = 2 nM T40556 CH1Y7G 132010677 Ki = 0.6 nM T40556 CJ2I1C 132010719 Ki = 0.5 nM T40556 C8IAW3 132010913 Ki = 1.5 nM T40556 CHO97Q 132010929 Ki = 1.3 nM T40556 CE61QG 132154358 IC50 = 0.43 nM T40556 COE15M 132166121 IC50 = 5100 nM T40556 CGNQ49 132168874 IC50 = 19000 nM T40556 CHC6A0 132168907 IC50 = 12000 nM T40556 CRV1I6 132168917 IC50 = 3800 nM T40556 CB4X0G 132169005 IC50 = 8900 nM T40556 CX9U1Y 132169030 IC50 > 20000 nM T40556 CO7QW0 132169133 IC50 = 7800 nM T40556 CD8SE7 132169397 IC50 > 20000 nM T40556 CG4X6Z 132169416 IC50 = 14000 nM T40556 CV8F3O 132169466 IC50 > 20000 nM T40556 C7EHB4 132169581 IC50 = 7400 nM T40556 CI3HC8 132169624 IC50 = 12000 nM T40556 CF7H3C 132169928 IC50 = 6900 nM T40556 C7KUC2 132176755 IC50 > 20000 nM T40556 C6HQ0I 132181409 IC50 > 20000 nM T40556 C2S4IT 132181414 IC50 = 1100 nM T40556 C3MV7Y 132181499 IC50 = 3900 nM T40556 CM2K6Z 132181651 IC50 = 18000 nM T40556 CZW36J 132181706 IC50 > 20000 nM T40556 CVZ87Y 132181707 IC50 = 4100 nM T40556 CXVW94 132181717 IC50 > 20000 nM T40556 CG13LT 132186451 IC50 = 15000 nM T40556 CGC84J 132186467 IC50 > 20000 nM T40556 CB23YA 132186468 IC50 = 8500 nM T40556 C06KYU 132186469 IC50 = 3200 nM T40556 CI56DE 132186470 IC50 > 20000 nM T40556 COK17B 132186514 IC50 = 14000 nM T40556 CE3H2T 132186523 IC50 = 2500 nM T40556 CG5SN9 132186583 IC50 = 4700 nM T40556 CN90OX 132186586 IC50 = 14000 nM T40556 CAR2X5 132186700 IC50 = 2800 nM T40556 C5A3QS 132186701 IC50 = 3300 nM T40556 CKY07I 132186706 IC50 > 20000 nM T40556 C4DOU1 132186760 IC50 > 20000 nM T40556 CFB2X6 132186767 IC50 = 13000 nM T40556 CM6K0J 132186772 IC50 = 7700 nM T40556 CL29US 132186773 IC50 = 11000 nM T40556 CUH7W8 132186890 IC50 = 6700 nM T40556 CGDN94 132275066 IC50 = 12000 nM T40556 C5LQ2Y 132289425 IC50 = 2511.89 nM T40556 CL1FY9 132451787 IC50 = 5600 nM T40556 C9UGN7 132503236 IC50 = 2700 nM T40556 CN3P0M 132961531 IC50 = 76 nM T40556 CU0E6V 132992936 IC50 = 234.42 nM T40556 C51OUR 133053976 IC50 = 52 nM T40556 C16VTU 134132238 IC50 > 20000 nM T40556 C6V4WU 134132252 IC50 = 9800 nM T40556 C5SV3A 134132771 IC50 > 20000 nM T40556 CANC79 134133805 IC50 > 20000 nM T40556 CAI3J0 134134171 IC50 = 18000 nM T40556 CFZ94S 134135176 IC50 = 7700 nM T40556 CV7K2Z 134135271 IC50 > 20000 nM T40556 C9OC2T 134135428 IC50 = 7420 nM T40556 C26RIB 134135696 IC50 = 4600 nM T40556 C8SCT7 134137178 IC50 > 20000 nM T40556 C7RFZ1 134139020 IC50 = 5800 nM T40556 C72VXC 134140106 IC50 = 6250 nM T40556 COC34Y 134140792 IC50 = 8240 nM T40556 CE16SF 134142067 IC50 > 20000 nM T40556 CU1Y5M 134142603 IC50 = 2740 nM T40556 C8D3NS 134143236 IC50 = 11000 nM T40556 CY83MP 134143286 IC50 > 20000 nM T40556 C1NKU6 134144625 IC50 = 11230 nM T40556 C1KAR7 134146622 IC50 > 20000 nM T40556 CWZ0V3 134147360 IC50 > 20000 nM T40556 CC87ZT 134149739 IC50 > 20000 nM T40556 CA2HB7 134149861 IC50 > 20000 nM T40556 CF98TY 134149949 IC50 > 20000 nM T40556 CC29GZ 134151635 IC50 > 20000 nM T40556 CP51GS 134151910 IC50 > 20000 nM T40556 CIP61L 134153498 IC50 = 37000 nM T40556 C31JZR 134154313 IC50 > 20000 nM T40556 COX6Y9 134157699 IC50 = 14000 nM T40556 CBW6T0 134163707 IC50 = 283 nM T40556 CO3A0E 134817551 IC50 = 5011.87 nM T40556 CP4X5W 134817552 IC50 = 5011.87 nM T40556 CS7WX6 134821995 IC50 = 1000 nM T40556 CI2AM1 134828588 IC50 = 100 nM T40556 CJ9E8M 135121918 IC50 = 70 nM T40556 CS71IF 135126189 IC50 = 280 nM T40556 CK1BA5 135126537 IC50 = 2600 nM T40556 CRS95D 135126542 IC50 = 970 nM T40556 CZQ49P 135126546 IC50 = 520 nM T40556 CTO4K5 135143907 IC50 = 3900 nM T40556 CIAG86 135394452 IC50 > 20000 nM T40556 CRNY32 135397673 Ki = 0.5 nM T40556 C9J4PW 135398123 IC50 = 1990 nM T40556 C7L5ER 135398124 IC50 = 690 nM T40556 C9IGU4 135398125 IC50 = 630 nM T40556 CCTO31 135404086 IC50 = 4300 nM T40556 C39LZE 135404087 IC50 = 5200 nM T40556 CA40QW 135535536 IC50 > 50118.72 nM T40556 CV4X7R 135566898 Ki = 910 nM T40556 CU2F1G 135566900 Ki = 150 nM T40556 C5F3LV 135567026 IC50 = 430 nM T40556 CF8TQ2 135567084 IC50 = 1160 nM T40556 CZ84OQ 135567317 Ki = 10 nM T40556 CV2YA3 135630716 IC50 = 16000 nM T40556 CZK84G 135630721 IC50 = 31000 nM T40556 CKD1O7 135804260 IC50 = 4700 nM T40556 C4DMZ9 136002815 Ki = 6430 nM T40556 C6HJ9W 136174597 Ki = 6480 nM T40556 C0AY8G 136174600 Ki = 6830 nM T40556 CX9IM7 136174601 Ki = 520 nM T40556 CB26GV 136174603 Ki = 1300 nM T40556 CY4G3S 136174604 Ki = 1270 nM T40556 CQ02PC 136174605 Ki = 4670 nM T40556 CFH95M 136174610 Ki = 500 nM T40556 C4BO0T 136174611 Ki = 2790 nM T40556 CG9N5D 136174612 Ki = 1400 nM T40556 C69HZF 136174618 Ki = 7140 nM T40556 CWSG57 136212224 IC50 = 4310 nM T40556 C41NGO 136224170 Ki = 1280 nM T40556 CL7FQ1 136224171 Ki = 2310 nM T40556 C7O5PH 136226498 Ki = 4920 nM T40556 C1RH2I 136226499 Ki = 5970 nM T40556 CHY5I0 136226500 Ki > 100000 nM T40556 CYVZ61 136226501 Ki = 7120 nM T40556 CXJG97 136226502 Ki = 6130 nM T40556 CBHW80 136226503 Ki = 900 nM T40556 CWD47H 136226504 Ki = 320 nM T40556 CKPS21 136226505 Ki = 730 nM T40556 CP29FE 136226506 Ki = 6540 nM T40556 C81XIB 136226507 Ki = 9600 nM T40556 C9OJ6K 136226508 Ki = 1300 nM T40556 C6JRN2 136226509 Ki = 1840 nM T40556 CNT61S 136226510 Ki = 3130 nM T40556 CW94QO 136226511 Ki = 169.82 nM T40556 CAFU62 136226512 Ki = 6020 nM T40556 CFT26V 136226513 Ki = 2390 nM T40556 CJG3I4 136226514 Ki = 3910 nM T40556 C2PB9D 136242352 IC50 = 560 nM T40556 C27WOL 136244604 IC50 = 77000 nM T40556 CW8XN5 136321792 IC50 = 9280 nM T40556 CXLE13 136387525 Ki = 30 nM T40556 CFRV40 136387526 Ki = 37 nM T40556 CSPK74 136387543 Ki = 16 nM T40556 C4N2FR 136387545 Ki = 77 nM T40556 CY3UK2 136387556 Ki = 1100 nM T40556 CL6R5U 136387567 Ki = 150 nM T40556 C53FKI 136577469 IC50 = 6380 nM T40556 C0IY2P 136963109 IC50 < 100 nM T40556 C60DNA 137250528 IC50 = 11000 nM T40556 C6G9UA 137275811 IC50 = 328 nM T40556 CO71RI 137285009 IC50 = 32 nM T40556 CS9MR6 137285011 IC50 = 32 nM T40556 CL02HM 137319656 IC50 = 2092 nM T40556 C5E8GX 137319657 IC50 = 1416 nM T40556 CI1WA0 137319664 IC50 = 6600 nM T40556 C6ZG7K 137321201 IC50 = 501.19 nM T40556 CFXE14 137321203 IC50 = 50.12 nM T40556 CXN4U1 137321204 IC50 = 63.1 nM T40556 C6MGN1 137322665 IC50 = 32230 nM T40556 C31BFH 137347775 IC50 = 540 nM T40556 C7FVC0 137347776 IC50 = 260 nM T40556 CG8VK6 137348598 IC50 = 2000 nM T40556 CMF86O 137348600 IC50 = 24000 nM T40556 CW1IF3 137348845 IC50 = 22000 nM T40556 C4VNB8 137369426 IC50 = 45 nM T40556 CTM7U5 137628634 IC50 = 45 nM T40556 CS6U7Y 137631402 IC50 = 720 nM T40556 C53KAO 137631500 IC50 = 4900 nM T40556 CU49YR 137631543 IC50 > 10000 nM T40556 COP3H7 137631627 IC50 = 120 nM T40556 CA2VS4 137631629 IC50 = 3900 nM T40556 C0Y3UF 137631784 IC50 = 10100 nM T40556 CNZS84 137631821 IC50 > 10000 nM T40556 CUE7F1 137631875 IC50 = 490 nM T40556 CR5FO2 137632087 Ki > 40000 nM T40556 C25OZB 137632559 IC50 > 20000 nM T40556 C7F4MJ 137632577 Ki = 190 nM T40556 CA2D8W 137632690 Ki > 40000 nM T40556 C5JP8O 137633986 IC50 = 12 nM T40556 CF9I7B 137634124 IC50 = 170 nM T40556 CYU6T2 137634563 IC50 > 20000 nM T40556 CX9OI0 137634784 IC50 = 180 nM T40556 C9XVL1 137635109 IC50 = 11200 nM T40556 CS27YB 137635150 IC50 = 401 nM T40556 CM9P2A 137635443 IC50 = 2300 nM T40556 CQW04U 137635588 Ki = 8.7 nM T40556 CBX4I3 137635735 IC50 = 530 nM T40556 C0D1LR 137635790 IC50 > 20000 nM T40556 CO0UN6 137635792 IC50 = 1500 nM T40556 CWYU04 137635881 IC50 > 10000 nM T40556 C2P8AM 137636088 Ki = 9 nM T40556 CQT3A9 137636309 IC50 > 100000 nM T40556 CYZJ80 137636683 IC50 = 4900 nM T40556 CO08EU 137636712 Ki = 2500 nM T40556 CCAP49 137636933 IC50 > 20000 nM T40556 C92AIX 137637032 Ki = 26 nM T40556 C69BGA 137637084 IC50 = 2470 nM T40556 C7NZ4E 137637179 IC50 = 3200 nM T40556 C05CVD 137637565 IC50 = 520 nM T40556 C1AB7Q 137637710 IC50 > 10000 nM T40556 CT2D8X 137638314 IC50 = 13000 nM T40556 CRN21V 137638824 IC50 = 1500 nM T40556 CVK32T 137639306 Ki = 160 nM T40556 C6ZG0E 137639443 IC50 = 160 nM T40556 CP2HK4 137639600 IC50 = 3800 nM T40556 CV1EP8 137639742 IC50 = 37000 nM T40556 CFS67E 137640120 IC50 = 1810 nM T40556 C5MS7I 137640141 IC50 = 40 nM T40556 CKUX65 137640422 IC50 = 6400 nM T40556 CF42ZW 137640560 IC50 = 8590 nM T40556 CJG6R8 137640750 IC50 = 3400 nM T40556 C0SYB2 137640929 IC50 = 18400 nM T40556 CL4FK6 137641456 IC50 > 20000 nM T40556 COK20S 137641504 IC50 = 1400 nM T40556 CXH59O 137641530 IC50 > 10000 nM T40556 C01BVT 137642411 IC50 = 2000 nM T40556 CMX9U6 137642634 IC50 > 10000 nM T40556 COY3A6 137642659 IC50 = 9200 nM T40556 C9XZ3O 137643020 IC50 = 2700 nM T40556 CGE1L2 137643245 Ki = 430 nM T40556 C41QFV 137643280 IC50 > 10000 nM T40556 C36RVQ 137643517 IC50 > 10000 nM T40556 CP28JU 137643679 IC50 > 10000 nM T40556 CD8VQ1 137643820 Ki > 40000 nM T40556 CDK90I 137643908 IC50 < 50 nM T40556 CQ0YM6 137643978 IC50 = 2200 nM T40556 CZXP42 137644405 IC50 > 20000 nM T40556 CRJ2W3 137644677 IC50 = 630 nM T40556 C2T8WQ 137644823 IC50 = 18500 nM T40556 C7G3SF 137644942 IC50 = 640 nM T40556 CYBP84 137644977 IC50 = 200 nM T40556 C37MBU 137645618 IC50 > 10000 nM T40556 CTG91Q 137646067 IC50 = 320 nM T40556 C0R3FG 137646519 IC50 = 4200 nM T40556 CGQ3X2 137647012 IC50 = 68 nM T40556 CWJ7N5 137647079 IC50 = 6900 nM T40556 CJ9UI7 137647118 IC50 > 20000 nM T40556 CXD50J 137647775 IC50 = 16800 nM T40556 CGX65O 137647885 IC50 > 20000 nM T40556 C2HTJ9 137648078 IC50 = 180 nM T40556 C8QO2D 137648257 Ki = 110 nM T40556 C6AXY7 137648298 IC50 = 17 nM T40556 CK16RO 137648883 IC50 = 5700 nM T40556 CV3J1C 137648959 IC50 > 10000 nM T40556 C9TC6G 137648962 Ki = 4.4 nM T40556 C0NR8F 137649215 IC50 = 130 nM T40556 C89VWP 137649346 IC50 = 6000 nM T40556 CQ9G8P 137649425 IC50 > 10000 nM T40556 CC2V9L 137649517 IC50 < 5 nM T40556 CA0G8B 137649726 IC50 < 50 nM T40556 C85QNS 137649815 IC50 = 9400 nM T40556 CKN60B 137649822 IC50 > 120000 nM T40556 CO7K6Y 137649906 IC50 = 13200 nM T40556 CZ4VH1 137650214 IC50 = 17 nM T40556 CM6S0X 137650255 IC50 > 20000 nM T40556 CQ5WF3 137650342 IC50 = 225 nM T40556 CM1WG7 137650502 IC50 = 3.1 nM T40556 CC34KQ 137650533 IC50 = 4600 nM T40556 CLGI76 137650651 IC50 > 10000 nM T40556 C4Y8HV 137650663 IC50 = 4600 nM T40556 C52APO 137650788 IC50 = 1530 nM T40556 C6FXI4 137650878 IC50 = 6370 nM T40556 CY0G4J 137650944 IC50 = 1040 nM T40556 CE42GP 137650954 IC50 = 4100 nM T40556 CSV15U 137650957 IC50 = 52000 nM T40556 C8UT7D 137651043 Ki = 460 nM T40556 C1MA2K 137651137 IC50 > 20000 nM T40556 CV9F6J 137651164 IC50 > 120000 nM T40556 C5Y0DH 137651263 IC50 > 20000 nM T40556 C2SMF1 137651591 Ki = 370 nM T40556 C6SKI2 137651884 IC50 > 20000 nM T40556 CHN7A8 137652035 IC50 = 4500 nM T40556 CMYI27 137652124 IC50 = 7400 nM T40556 CG9OR2 137652284 IC50 > 10000 nM T40556 C82CEA 137652287 IC50 = 36 nM T40556 CB3J9E 137652309 IC50 = 25000 nM T40556 C5ANC9 137652708 IC50 = 430 nM T40556 CCZD32 137652808 IC50 = 9400 nM T40556 CT17HB 137653121 Ki = 2200 nM T40556 CHU2W4 137653154 IC50 > 120000 nM T40556 CM9HL5 137653223 IC50 = 140 nM T40556 CA4WO8 137653484 Ki = 140 nM T40556 C7Y6IH 137653562 IC50 = 4300 nM T40556 C7APB1 137653732 IC50 = 3240 nM T40556 CL1V9T 137654008 IC50 = 4400 nM T40556 C7G8AR 137654107 IC50 = 490 nM T40556 CZ1K6N 137654718 Ki = 10000 nM T40556 C3OX9R 137655043 IC50 > 10000 nM T40556 C7L6MV 137655172 IC50 > 20000 nM T40556 CVH74T 137655200 Ki = 1200 nM T40556 CWPO58 137655523 IC50 = 1040 nM T40556 CGC79R 137655670 IC50 > 10000 nM T40556 CQ9UL6 137655871 IC50 = 390 nM T40556 CM7Y4D 137655923 IC50 = 13900 nM T40556 C5B7LO 137656022 IC50 = 5800 nM T40556 CX35DY 137656164 IC50 = 8300 nM T40556 C8BP5R 137656667 IC50 = 15000 nM T40556 C1SBT0 137656977 IC50 > 10000 nM T40556 CW9C8L 137657087 IC50 = 14400 nM T40556 C1YOL6 137657448 Ki = 100 nM T40556 C5TEY3 137657620 IC50 > 80000 nM T40556 C9LHE3 137657639 IC50 > 10000 nM T40556 C9DGJ2 137657716 Ki = 8.2 nM T40556 C1N7LY 137658279 IC50 > 20000 nM T40556 CE3CQ5 137659158 IC50 = 1600 nM T40556 CAS5V7 137659228 Ki = 3.4 nM T40556 C5TDP8 137660755 Ki = 3000 nM T40556 CT9Z7G 137661063 IC50 = 97 nM T40556 C7F1YH 137661082 IC50 = 9 nM T40556 CI6B7L 137661152 IC50 = 350 nM T40556 C3NPW0 137661190 IC50 = 200 nM T40556 C4XR7V 137661795 IC50 > 10000 nM T40556 C8TO4R 137662308 IC50 > 10000 nM T40556 CM3UF7 137700779 IC50 > 10000 nM T40556 CU5N8O 137701509 IC50 = 1700 nM T40556 CYV4O3 138756791 IC50 = 1300 nM T40556 CQ6XB7 139030526 IC50 = 19952.62 nM T40556 C1G9LA 139035062 Ki = 7.3 nM T40556 CPY8E7 139341516 IC50 = 10 nM T40556 COE12P 139341517 IC50 = 3600 nM T40556 C3HJI2 139341518 IC50 = 669 nM T40556 CWK82L 139341520 IC50 = 67.3 nM T40556 C3DGA7 139341522 IC50 = 11.7 nM T40556 C4CHN3 139341523 IC50 = 76 nM T40556 CRW7P5 139341524 IC50 = 9.5 nM T40556 C98TAG 139341527 IC50 = 15 nM T40556 CJ01EC 139341528 IC50 = 78.6 nM T40556 C5F7OS 139341530 IC50 > 1000 nM T40556 COY2D4 139341532 IC50 = 128 nM T40556 CVLH98 139341533 IC50 = 1600 nM T40556 C6BV5E 139341541 IC50 = 4.2 nM T40556 CWM81B 139341544 IC50 = 4.7 nM T40556 CF1VL4 139341553 IC50 = 117 nM T40556 CF8LU1 139341570 IC50 = 16.2 nM T40556 C3SVA5 139341572 IC50 = 3.5 nM T40556 CL9XU2 139341575 IC50 = 28.4 nM T40556 C69JHS 139341584 IC50 = 229 nM T40556 CJ9TL3 139341588 IC50 > 2000 nM T40556 C7IN1U 139341589 IC50 = 438 nM T40556 C0HT4J 139341591 IC50 = 97.9 nM T40556 CF2D6W 139341726 IC50 = 788 nM T40556 CI1H2T 139341727 IC50 = 740 nM T40556 C9K8YX 139341747 IC50 > 1000 nM T40556 C4YMW6 139341818 IC50 = 71.3 nM T40556 CYQ79A 139382567 IC50 > 20000 nM T40556 C24DCX 139547911 IC50 = 296 nM T40556 C0D6ZN 141531706 IC50 > 100 nM T40556 C1YV7C 141531707 IC50 > 100 nM T40556 C8ZQ2U 141736359 IC50 > 20000 nM T40556 C5VNM4 141736367 IC50 > 20000 nM T40556 C4H6ZE 141759312 IC50 = 930 nM T40556 CH0I8X 142296514 IC50 = 238.5 nM T40556 CR2UQ8 142296515 IC50 = 20.4 nM T40556 CDK17C 142296518 IC50 = 1470 nM T40556 C9U5OC 142296519 IC50 = 1350 nM T40556 C45FBX 142296520 IC50 = 350 nM T40556 CV01UW 142296521 IC50 = 54.6 nM T40556 C9F8QZ 142296524 IC50 = 125.5 nM T40556 C4B7JP 142296525 IC50 = 10.3 nM T40556 C12UVJ 142296527 IC50 = 1030 nM T40556 CAI65C 142296528 IC50 > 1000 nM T40556 CL56YI 142296532 IC50 = 730 nM T40556 C8I1XZ 142296533 IC50 = 10.5 nM T40556 C6BL0T 142296538 IC50 = 389 nM T40556 CB17LA 142296539 IC50 = 770 nM T40556 CJLX96 142296540 IC50 = 17.2 nM T40556 CNTR63 142296543 IC50 = 124.5 nM T40556 CCI89P 142296544 IC50 > 1000 nM T40556 C0AZR5 142296546 IC50 = 20.9 nM T40556 CH1DE5 142296549 IC50 = 320 nM T40556 CJGR35 142296552 IC50 = 22.3 nM T40556 C1O4EU 142296553 IC50 = 189.5 nM T40556 C8JD1T 142296555 IC50 = 31.3 nM T40556 CW5UI4 142296557 IC50 = 81.7 nM T40556 C9BGH7 142296560 IC50 = 73.8 nM T40556 CKR85F 142296562 IC50 = 62.3 nM T40556 CH5Q3R 142296563 IC50 = 175.8 nM T40556 C1IX7Q 142296567 IC50 = 46.4 nM T40556 C26QKE 142296568 IC50 = 1574.5 nM T40556 CU2FS3 142296570 IC50 = 27.4 nM T40556 CQV3X9 142296573 IC50 = 17.4 nM T40556 CT7NJ3 142296575 IC50 = 60.7 nM T40556 CH9UR4 142296576 IC50 = 760 nM T40556 CD8ZU4 142296577 IC50 = 380 nM T40556 C6VJQ4 142296579 IC50 = 199 nM T40556 C6N2KD 142296581 IC50 = 36.2 nM T40556 CM8D2W 142296582 IC50 = 20.2 nM T40556 C29URB 142296583 IC50 = 770 nM T40556 C7O2GC 142296584 IC50 = 1040 nM T40556 C9R8DG 142296585 IC50 = 357 nM T40556 CM51HE 142296589 IC50 = 13.6 nM T40556 CPC79Y 142296592 IC50 = 37.9 nM T40556 CX1F8A 142296595 IC50 = 10.6 nM T40556 CVZ0W4 142296596 IC50 = 270 nM T40556 CI73SX 142296601 IC50 = 285.5 nM T40556 C7VS9Z 142296602 IC50 = 250 nM T40556 CP2M0O 142296603 IC50 = 240 nM T40556 CW1FX5 142296604 IC50 = 177.5 nM T40556 CZSB40 142296605 IC50 = 152.5 nM T40556 CJAM56 142296607 IC50 = 15.9 nM T40556 CIWV81 142296611 IC50 = 1530 nM T40556 CG6X3A 142535938 EC50 = 526 nM T40556 CQB16E 142577810 IC50 = 398.11 nM T40556 CWYC72 142577823 IC50 = 398.11 nM T40556 CM3R1C 142577824 IC50 = 630.96 nM T40556 C6E2DB 142577846 IC50 = 316.23 nM T40556 C6X5VA 142577862 IC50 = 501.19 nM T40556 CWV83D 142577883 IC50 = 1258.93 nM T40556 C6YPL1 142740580 IC50 = 25.12 nM T40556 CWE84Z 142740586 IC50 = 39.81 nM T40556 CWHP86 142740595 IC50 = 79.43 nM T40556 C0WX3V 145829181 IC50 = 100 nM T40556 CXV80B 145829182 IC50 = 2479 nM T40556 CD6U7X 145925666 IC50 = 87.7 nM T40556 C8OD1K 145925690 IC50 = 165.96 nM T40556 C7EB9S 145945981 IC50 = 4.5 nM T40556 CR6V5X 145946095 IC50 = 12589.25 nM T40556 C0CE9F 145946096 IC50 = 6309.57 nM T40556 C25ZQV 145946097 IC50 = 251.19 nM T40556 C6VNJ7 145949319 IC50 = 510 nM T40556 CZ9U2C 145949385 IC50 = 270 nM T40556 C1CIP3 145949560 IC50 = 530 nM T40556 CS96DV 145950283 IC50 = 2120 nM T40556 C48MVS 145950376 IC50 = 2270 nM T40556 C1VM4D 145950404 IC50 = 18720 nM T40556 CUTA34 145950411 IC50 = 180 nM T40556 CH93SO 145950673 IC50 = 13300 nM T40556 CW58CR 145950888 IC50 = 610 nM T40556 C96NCH 145950955 IC50 > 20000 nM T40556 C21NAZ 145951567 IC50 = 170 nM T40556 C1XZG5 145951828 IC50 = 280 nM T40556 C1HLK5 145951928 IC50 = 17 nM T40556 CEA0I1 145952035 IC50 = 69230 nM T40556 C3ZV1O 145952497 IC50 > 20000 nM T40556 CRL42T 145953028 IC50 = 580 nM T40556 CNU28F 145953072 IC50 = 23060 nM T40556 C9I0SC 145953078 IC50 = 830 nM T40556 CVN8A5 145953287 IC50 = 620 nM T40556 CI9U2L 145953592 IC50 = 490 nM T40556 CC5D1Q 145953654 IC50 = 1330 nM T40556 CSR9N7 145953663 IC50 = 480 nM T40556 CBNI84 145953835 IC50 = 1170 nM T40556 C0ZTC4 145954129 IC50 = 110 nM T40556 C2MYA1 145954210 IC50 = 790 nM T40556 CTE74G 145954441 IC50 > 20000 nM T40556 CH14TJ 145954453 IC50 = 860 nM T40556 CBYF17 145954698 IC50 = 290 nM T40556 CR6OX1 145954766 IC50 = 120 nM T40556 CMCH58 145954903 IC50 = 13260 nM T40556 C6D0OT 145955789 IC50 > 20000 nM T40556 CMQ3J7 145955860 IC50 = 4250 nM T40556 CF0EK4 145956136 IC50 = 230 nM T40556 CB61VZ 145956237 IC50 = 270 nM T40556 C8M5DP 145956320 IC50 = 200 nM T40556 C8SC9E 145956329 IC50 = 3540 nM T40556 CIU29S 145956336 IC50 = 1140 nM T40556 CCNU52 145956492 IC50 = 570 nM T40556 C50CSO 145956910 IC50 = 180 nM T40556 CN5YO3 145957310 IC50 > 20000 nM T40556 CEJA84 145957398 IC50 = 50750 nM T40556 C9J2GS 145957453 IC50 > 20000 nM T40556 C42KZE 145957509 IC50 = 400 nM T40556 CIW97K 145957788 IC50 = 270 nM T40556 CSK9W5 145957886 IC50 = 520 nM T40556 CX7C4V 145958221 IC50 = 3640 nM T40556 CIDU52 145958263 IC50 = 340 nM T40556 C0IN8H 145958454 IC50 = 460 nM T40556 C7C5WL 145958595 IC50 = 2190 nM T40556 C2VNR7 145958596 IC50 = 290 nM T40556 C0CUF6 145958773 IC50 = 1170 nM T40556 CA9UQ0 145959024 IC50 > 1000 nM T40556 CT96GS 145959255 IC50 = 410 nM T40556 C30DFL 145959472 IC50 = 27520 nM T40556 CDNG83 145959505 IC50 = 150 nM T40556 C8AP9H 145959530 IC50 = 360 nM T40556 CIZW13 145959848 IC50 = 1430 nM T40556 C85NDV 145959886 IC50 = 6070 nM T40556 CGA86D 145960246 IC50 = 12710 nM T40556 C5R2OX 145960489 IC50 = 602.56 nM T40556 CR7Q6O 145960620 IC50 = 1230.27 nM T40556 C8DIH1 145960623 IC50 = 1100 nM T40556 CRPN57 145960718 IC50 = 585 nM T40556 CBC6Z8 145960723 IC50 = 2238.72 nM T40556 CG27BX 145961203 IC50 = 120 nM T40556 CL4XG1 145961395 IC50 = 793 nM T40556 CSDU51 145961590 IC50 = 842 nM T40556 CDZ8R4 145961700 IC50 = 722 nM T40556 CY2B3F 145961967 IC50 = 630.96 nM T40556 C90WEP 145961969 IC50 = 4680 nM T40556 C5PN9T 145962081 IC50 = 810 nM T40556 CJY05H 145962174 IC50 = 165.96 nM T40556 CKQ3G4 145962258 IC50 = 1412.54 nM T40556 CAF0K5 145962473 IC50 = 269.15 nM T40556 CEZ30H 145962475 IC50 = 4265.8 nM T40556 C49WON 145962542 IC50 = 489.78 nM T40556 C5T0KG 145962602 IC50 = 945 nM T40556 CBU2O7 145962767 IC50 = 478 nM T40556 C3YL0V 145962799 IC50 = 302 nM T40556 C6V3LN 145962814 IC50 = 3800 nM T40556 CMW3L6 145963581 IC50 = 380.19 nM T40556 CM4RN5 145963629 IC50 = 954.99 nM T40556 CH4QA2 145963723 IC50 = 3235.94 nM T40556 CC06PY 145963915 IC50 = 41900 nM T40556 CT3G0N 145963947 IC50 = 630.96 nM T40556 CU7WE5 145964377 Ki = 6.5 nM T40556 CC17DU 145964393 IC50 = 253 nM T40556 CH06LF 145964543 IC50 = 104 nM T40556 CT28NG 145964553 IC50 = 316.23 nM T40556 C4CIF7 145965008 IC50 = 794.33 nM T40556 C6EOB0 145965052 IC50 = 184.5 nM T40556 C72YHJ 145965062 Ki = 57 nM T40556 CD2WO6 145965211 IC50 = 5011.87 nM T40556 CCW5X8 145965219 IC50 = 107 nM T40556 C3FJ0L 145965372 IC50 = 100 nM T40556 CKNE25 145965382 IC50 = 251.19 nM T40556 C6M3FN 145965388 Ki = 17 nM T40556 CJ07ZP 145965402 IC50 = 125.89 nM T40556 C0X8PE 145965751 IC50 = 1000 nM T40556 CQC15M 145966021 IC50 = 79.43 nM T40556 CCTY08 145966026 IC50 = 107.5 nM T40556 C2Q7ES 145966038 IC50 = 100 nM T40556 CJ27UK 145966193 Ki < 0.5 nM T40556 CJ5BC4 145966522 IC50 = 2.3 nM T40556 C4ED6N 145966560 IC50 = 501.19 nM T40556 CE4D5F 145966579 IC50 = 596 nM T40556 C8XR2B 145966639 IC50 = 25118.86 nM T40556 C5BFX2 145966845 IC50 = 2511.89 nM T40556 CC05ZI 145967006 IC50 = 316.23 nM T40556 C4Y0PN 145967100 IC50 > 20000 nM T40556 C0T3BJ 145967243 IC50 = 1000 nM T40556 CYV74C 145967245 Ki = 10.5 nM T40556 C1V2DR 145967422 IC50 = 50.12 nM T40556 CHQ9L0 145967434 IC50 = 168 nM T40556 C2M7TI 145967443 IC50 = 370 nM T40556 CXWZ04 145967512 IC50 = 421 nM T40556 CX1C4W 145967999 IC50 = 4.3 nM T40556 CV4LN0 145968329 IC50 = 72000 nM T40556 C7SC5G 145968551 IC50 = 121000 nM T40556 CT06PA 145969741 IC50 = 15000 nM T40556 C9S8GB 145969777 IC50 > 200000 nM T40556 C0ZN2W 145969902 IC50 = 26000 nM T40556 C4YE5O 145970005 IC50 = 49000 nM T40556 CS6N3Y 145970287 IC50 > 10000 nM T40556 C13UOX 145970508 IC50 = 158.49 nM T40556 CO4RB3 145970920 IC50 = 24000 nM T40556 C7SK4T 145971247 IC50 > 1000 nM T40556 CDB65R 145971415 IC50 = 125.89 nM T40556 CCAT53 145971461 IC50 = 200 nM T40556 CF37MT 145971516 IC50 = 210 nM T40556 C3BSE8 145971523 IC50 = 590 nM T40556 C4GX3P 145971629 IC50 = 630.96 nM T40556 C9Q5RW 145971747 IC50 = 880 nM T40556 CV0TS2 145971844 IC50 = 794.33 nM T40556 CH8Y6A 145971920 IC50 = 1020 nM T40556 CIJO67 145972096 IC50 = 650 nM T40556 CV83ED 145972103 Ki = 1.2 nM T40556 C4D8RC 145972215 IC50 = 100 nM T40556 C0PFQ7 145972286 IC50 > 10000 nM T40556 CN70KV 145972360 IC50 = 95 nM T40556 CNU4O9 145972623 IC50 = 5100 nM T40556 C2RTO8 145972845 IC50 = 107 nM T40556 CQ35BN 145972969 IC50 = 1258.93 nM T40556 CD4A3Y 145973334 IC50 > 20000 nM T40556 C1Z3WQ 145973981 IC50 = 794.33 nM T40556 CWQ6A5 145974124 Ki = 2.7 nM T40556 CP49HN 145974181 IC50 > 20000 nM T40556 CXF6B5 145974721 IC50 = 501.19 nM T40556 CW37DI 145974796 IC50 = 87 nM T40556 CE7O2Z 145974859 Ki < 0.5 nM T40556 CG0D7U 145974979 IC50 = 100 nM T40556 CA85TK 145975493 IC50 > 20000 nM T40556 C6R2YM 145975649 IC50 = 2579 nM T40556 CTAZ41 145975701 IC50 > 50000 nM T40556 CW56PH 145975703 IC50 = 28 nM T40556 CRZ78W 145975795 IC50 = 630.96 nM T40556 CH57GW 145975937 IC50 = 186 nM T40556 CN4O0K 145976012 IC50 = 310 nM T40556 CKG83I 145976334 Ki = 641 nM T40556 CG0ZO6 145976380 IC50 = 794.33 nM T40556 CAL91V 145976398 IC50 = 158.49 nM T40556 CS05DX 145976415 IC50 = 1584.89 nM T40556 CR28YS 145976646 IC50 = 59 nM T40556 C26XFE 145976805 IC50 = 158.49 nM T40556 C1F7DT 145976814 IC50 = 398.11 nM T40556 C7J1IZ 145976831 IC50 = 168 nM T40556 CVJ61U 145977109 IC50 = 690 nM T40556 C3NUY9 145977309 Ki = 2.7 nM T40556 COD4I9 145977320 IC50 = 199.53 nM T40556 CG5TD0 145977365 IC50 = 63.1 nM T40556 C6M2CY 145977402 IC50 = 1258.93 nM T40556 CX13RH 145977417 IC50 = 1258.93 nM T40556 C63KPH 145977495 IC50 = 630.96 nM T40556 CB9F1X 145977980 IC50 = 94 nM T40556 C0MD9U 145978238 IC50 = 183 nM T40556 CJE53V 145978248 Ki = 7.7 nM T40556 C6S9BA 145978560 IC50 = 501.19 nM T40556 CSKC69 145978686 IC50 = 794.33 nM T40556 C8CO6S 145978782 IC50 = 50.12 nM T40556 C3LC2N 145978789 Ki = 4.4 nM T40556 CK4PH5 145978839 IC50 = 1108.5 nM T40556 CXC9E4 145978854 IC50 = 63.1 nM T40556 C0AI4C 145979130 IC50 = 25430 nM T40556 CAV7J5 145979375 IC50 = 1440 nM T40556 CV4TW9 145979405 IC50 = 6 nM T40556 CY6S4Z 145979516 IC50 = 4790 nM T40556 CYZ14K 145979939 IC50 = 12010 nM T40556 CHM8L7 145981045 IC50 = 1995.26 nM T40556 C9AUV1 145981148 IC50 = 630.96 nM T40556 CVYU19 145981267 IC50 = 2960 nM T40556 CJ0T1R 145981696 IC50 = 3870 nM T40556 CRXH81 145981836 IC50 = 794.33 nM T40556 CI5H7L 145982424 IC50 = 4730 nM T40556 CJ3FL8 145982835 IC50 > 50118.72 nM T40556 CA2W8M 145984295 IC50 = 31622.78 nM T40556 C4HWL1 145984406 IC50 = 40100 nM T40556 CE05ZV 145984432 IC50 = 25118.86 nM T40556 CV4GH7 145984467 IC50 = 7943.28 nM T40556 CT6V0I 145985751 IC50 = 6309.57 nM T40556 C0GHY5 145986052 IC50 = 158489.32 nM T40556 C69GXS 145986370 IC50 = 25118.86 nM T40556 C3OS2V 145987227 IC50 > 50000 nM T40556 C3QEX7 145987948 IC50 = 81000 nM T40556 CK20BY 145988169 Ki = 152 nM T40556 CY0OK3 145988346 IC50 = 794.33 nM T40556 CHL20Z 145988638 IC50 > 50000 nM T40556 COZ5J9 145989122 IC50 = 5011.87 nM T40556 COC35Q 145989187 IC50 = 501.19 nM T40556 CN4HR9 145989400 IC50 = 4770 nM T40556 CKP14Z 145989459 IC50 > 50000 nM T40556 C0NHS8 145989546 IC50 > 50000 nM T40556 CGY12F 145989646 IC50 = 2730 nM T40556 C7WRS3 145989682 IC50 = 2 nM T40556 CC9OS3 145989699 IC50 = 630.96 nM T40556 CC6NH9 145989855 IC50 = 1584.89 nM T40556 CSF47C 145990617 IC50 = 9320 nM T40556 CM5N9Y 145991689 IC50 = 1000 nM T40556 CSG40R 145991750 IC50 > 50000 nM T40556 C1SQD3 145992400 IC50 = 3590 nM T40556 CSN3C8 145992593 IC50 = 501.19 nM T40556 C1DP4O 146027046 Ki = 1.1 nM T40556 CK98QJ 146035912 IC50 > 50118.72 nM T40556 C53GZM 146037608 IC50 = 130 nM T40556 CZY8D7 146037609 IC50 = 2700 nM T40556 CL9TB0 146037610 IC50 > 10000 nM T40556 CBRE71 146047136 IC50 = 2.6 nM T40556 C3XOR2 146322224 IC50 = 6.1 nM T40556 C9TW5Q 146322225 IC50 = 100.4 nM T40556 CR12JW 146322226 IC50 = 7.9 nM T40556 CGV47C 146322227 IC50 = 9.6 nM T40556 CAE39T 146322229 IC50 = 8.7 nM T40556 CZ5KA1 146322241 IC50 = 142 nM T40556 CI2HL1 146322248 IC50 = 5.2 nM T40556 CQF42T 146322251 IC50 = 9.4 nM T40556 CH1I3X 146322264 IC50 = 4.2 nM T40556 C8LXY6 146322265 IC50 = 8.6 nM T40556 C3MT7G 146322268 IC50 = 5.9 nM T40556 C3R5OK 146322269 IC50 = 4.6 nM T40556 CJO2X3 146322270 IC50 = 5.3 nM T40556 CQ0S8V 146322271 IC50 = 7 nM T40556 CQG82Z 146322272 IC50 = 4.8 nM T40556 CC6RE8 146322280 IC50 = 4.6 nM T40556 C1G3IC 146322281 IC50 = 6.6 nM T40556 CFV96I 146322282 IC50 = 27.2 nM T40556 C4WYD7 146322283 IC50 = 6.8 nM T40556 C3QPV4 146322290 IC50 = 5.4 nM T40556 CG50HD 146322292 IC50 = 7.1 nM T40556 C2XWK6 146322293 IC50 = 5.8 nM T40556 CT6XO0 146322294 IC50 = 5.7 nM T40556 CZ3T7Q 146322295 IC50 = 14.4 nM T40556 C2ZVK5 146322296 IC50 = 9.5 nM T40556 CLK37M 147133615 Ki = 54.4 nM T40556 CTQ01S 147823626 Ki = 736 nM T40556 COU42L 147881243 IC50 = 92 nM T40556 CGW0K7 148225107 Ki = 376 nM T40556 CPQ57V 148251486 IC50 = 39.6 nM T40556 C5O7VJ 148648403 Ki = 50.3 nM T40556 CIUR70 149201098 Ki = 102 nM T40556 CWG10H 151364732 IC50 = 1190 nM T40556 CP5V2U 152625752 IC50 = 9.7 nM T40556 C6I7OZ 152636346 IC50 = 980 nM T40556 C7LM4U 153534003 IC50 = 1930 nM T40556 CP1V9H 153534004 IC50 = 1770 nM T40556 C9FIY4 153534005 IC50 = 710 nM T40556 CVT63S 153534008 IC50 = 2190 nM T40556 CZCD51 155352257 IC50 = 3900 nM T40556 CM4V9L 155352262 IC50 = 11000 nM T40556 C40KOR 155352277 IC50 > 100000 nM T40556 CZ50CJ 155352280 IC50 = 4500 nM T40556 C5K3FL 155352284 IC50 > 100000 nM T40556 CG6HY5 155352290 IC50 > 100000 nM T40556 C1ZFB8 155352296 IC50 > 100000 nM T40556 CPZ64D 155352301 IC50 = 1700 nM T40556 CB8EF6 155352304 IC50 = 61000 nM T40556 C02EIO 155352320 IC50 > 100000 nM T40556 C40RYV 155352344 IC50 > 100000 nM T40556 CHG13B 155352345 IC50 = 9700 nM T40556 CFD6H1 155352361 IC50 = 75000 nM T40556 CL2ZE0 155352369 IC50 > 100000 nM T40556 C8GZL5 155352384 IC50 = 1300 nM T40556 CFK2B1 155352401 IC50 = 102000 nM T40556 C0RO5V 155352412 IC50 = 12000 nM T40556 CZ1A8M 155352425 IC50 = 97000 nM T40556 C7U0VB 155352430 IC50 = 27000 nM T40556 C9FR3V 155510506 IC50 = 5930 nM T40556 CPY92M 155510533 IC50 = 310 nM T40556 CLMX96 155510847 Ki = 1 nM T40556 C2CD3Y 155510879 IC50 = 5540 nM T40556 CQUC76 155510893 Ki = 92 nM T40556 C98HOQ 155511096 Ki = 0.5 nM T40556 C9AXU3 155511227 IC50 = 169.1 nM T40556 CI6SA1 155511268 Ki = 945 nM T40556 CO0B1A 155511836 IC50 = 1529 nM T40556 C3R1EO 155511887 Ki = 15.85 nM T40556 C0LH8C 155511921 IC50 > 10000 nM T40556 C2D1SB 155512075 IC50 = 10000 nM T40556 CT2H3S 155512097 IC50 = 3100 nM T40556 CF6S3U 155512187 IC50 = 223 nM T40556 CD3LA9 155512613 IC50 > 50118.72 nM T40556 C51DIZ 155512733 IC50 = 62 nM T40556 C76QMK 155513141 Ki = 14.8 nM T40556 C5WUJ6 155513192 IC50 > 10000 nM T40556 C1D6MT 155513275 Ki = 50.12 nM T40556 CNQ9S2 155513363 IC50 = 205.2 nM T40556 CG47KU 155513649 Ki = 20 nM T40556 C9IUC2 155513805 IC50 = 1790 nM T40556 CF0GQ6 155513971 IC50 = 501.19 nM T40556 CP6VY4 155514289 Ki = 13 nM T40556 CI5CW6 155514299 Ki = 3.2 nM T40556 CS65YK 155514303 IC50 = 10 nM T40556 CH9KM8 155514491 IC50 = 655.8 nM T40556 C5JMW2 155514540 IC50 = 68 nM T40556 CNSC23 155514584 IC50 = 10 nM T40556 C30COX 155514594 IC50 = 6300 nM T40556 C27LFN 155514936 IC50 = 560 nM T40556 CX5W9H 155515117 IC50 = 5000 nM T40556 CE13CA 155515130 IC50 > 50118.72 nM T40556 C4THO2 155515131 Ki = 9.6 nM T40556 CH0LR3 155515173 IC50 = 50 nM T40556 CZU79I 155515498 IC50 = 6740 nM T40556 C8NC6V 155515565 IC50 = 8 nM T40556 C4GEL0 155515650 Ki = 18 nM T40556 CT03IV 155516089 IC50 = 1569 nM T40556 CZYP31 155516103 Ki = 1.3 nM T40556 C2GB7R 155516112 IC50 = 54 nM T40556 CPM43N 155516232 IC50 > 50118.72 nM T40556 CTI9Q6 155516388 IC50 = 19006 nM T40556 CNCH70 155516682 Ki = 1.1 nM T40556 CX6N4Z 155516719 IC50 = 1584.89 nM T40556 CDCH75 155516938 IC50 = 2598 nM T40556 CT5ZC6 155516968 IC50 = 22 nM T40556 C23BXS 155517049 IC50 > 50118.72 nM T40556 CP3K4R 155517232 IC50 = 44 nM T40556 CF0C7V 155517447 IC50 = 20.9 nM T40556 CS28LW 155517521 Ki = 47.3 nM T40556 CE0CX6 155517720 IC50 = 3466 nM T40556 C6Q3JK 155517968 IC50 > 50118.72 nM T40556 C8HK5X 155518008 IC50 = 1000 nM T40556 C32FEU 155518033 IC50 = 163.7 nM T40556 CFP24B 155518498 IC50 = 15848.93 nM T40556 CGBZ95 155518530 IC50 = 17.4 nM T40556 CBM34J 155518876 Ki = 3.162 nM T40556 CP2T0H 155519067 Ki = 413 nM T40556 C2GN1Y 155519159 IC50 = 5600 nM T40556 CHP0T5 155519310 IC50 = 10 nM T40556 C5KZG7 155519527 IC50 = 73 nM T40556 CW4HJ7 155519805 IC50 = 12.6 nM T40556 C8NL9U 155519897 IC50 = 140 nM T40556 CFVU05 155519921 IC50 = 480 nM T40556 C1JT3F 155520065 IC50 = 91.3 nM T40556 CY0A8O 155520236 IC50 = 167.1 nM T40556 CMVW63 155520501 IC50 = 37 nM T40556 C95RHU 155520664 IC50 = 1500 nM T40556 CGUX31 155520762 IC50 = 6680 nM T40556 CSPY94 155520847 Ki = 1.8 nM T40556 CB49NL 155521254 IC50 = 12589.25 nM T40556 C7UKD6 155521295 Ki = 617 nM T40556 C5F1JC 155521775 IC50 = 6020 nM T40556 CC30UG 155521851 IC50 > 50118.72 nM T40556 CAL9J8 155521991 IC50 = 1130 nM T40556 CH14KR 155522315 IC50 = 6000 nM T40556 CP9VQ4 155522638 Ki = 15 nM T40556 C0SE4F 155522830 Ki = 3.7 nM T40556 C0AP3M 155522854 IC50 < 1.995 nM T40556 C30NMB 155523002 IC50 = 1645 nM T40556 CHG5N8 155523095 IC50 > 10000 nM T40556 C85RSC 155523105 Ki = 92.6 nM T40556 CH06TJ 155523190 Ki = 25 nM T40556 CJYZ12 155523212 IC50 = 205.2 nM T40556 CL1P4M 155523233 IC50 > 50118.72 nM T40556 C1LK5T 155523560 Ki = 0.7 nM T40556 C1W8JL 155523577 IC50 > 50118.72 nM T40556 C2K9NI 155523694 IC50 > 50118.72 nM T40556 C8U2FI 155523758 Ki = 0.9 nM T40556 C0VS8H 155523850 IC50 > 50118.72 nM T40556 C3NYK0 155523937 IC50 = 50118.72 nM T40556 CBPV08 155523967 IC50 = 13120 nM T40556 CB90JU 155524196 IC50 = 11400 nM T40556 C2V0OA 155524426 IC50 = 265.6 nM T40556 CXM7E8 155524802 Ki = 80.6 nM T40556 C5BX4C 155525302 IC50 = 1250 nM T40556 C7GQN6 155525350 IC50 = 251.19 nM T40556 CSN27B 155525408 Ki = 22 nM T40556 CJ0V6I 155525482 Ki = 7.943 nM T40556 CW8O7G 155525483 IC50 > 50118.72 nM T40556 CF2P9Y 155525718 IC50 = 2100 nM T40556 CH79NC 155526096 IC50 = 125.89 nM T40556 C9I2LV 155526120 IC50 = 1400 nM T40556 CO1S0P 155526228 IC50 = 22700 nM T40556 C3QV1O 155526357 Ki = 9.5 nM T40556 C6R9LD 155526395 Ki = 66 nM T40556 CRK6E2 155526401 IC50 = 794.33 nM T40556 CKD9U4 155526975 IC50 = 3200 nM T40556 CVY04U 155527380 IC50 = 13000 nM T40556 C54DZA 155527566 IC50 = 1600 nM T40556 COY9L2 155527786 IC50 = 3724 nM T40556 CK2W1L 155527824 IC50 = 36 nM T40556 C43ZEI 155527951 IC50 = 501.19 nM T40556 CV7G8W 155527989 Ki = 5.012 nM T40556 C7Y5HX 155527993 IC50 = 1810 nM T40556 CLY27Z 155528197 Ki = 1.1 nM T40556 COJ86W 155528199 Ki = 0.7 nM T40556 CX18IT 155528305 IC50 = 1696 nM T40556 CKR6V3 155528325 IC50 > 50118.72 nM T40556 C3P9LB 155528627 Ki = 63.1 nM T40556 CEVB10 155528780 IC50 = 1900 nM T40556 CV7I6Z 155528992 IC50 = 53.8 nM T40556 C7MC0H 155529162 Ki = 68.4 nM T40556 COX8K5 155529510 IC50 > 50118.72 nM T40556 CIV12T 155529744 IC50 = 9930 nM T40556 CVMC06 155529991 IC50 > 50118.72 nM T40556 CO6X5T 155530144 IC50 = 16.6 nM T40556 CL93CM 155530154 IC50 > 50118.72 nM T40556 CQ2U3P 155530217 IC50 = 299.3 nM T40556 CEI09V 155530332 IC50 = 19952.62 nM T40556 CMSW35 155530439 IC50 = 1995.26 nM T40556 C2Y1DU 155530564 IC50 = 37.5 nM T40556 CY7ST9 155530616 IC50 > 50118.72 nM T40556 CB5Z9W 155530732 IC50 = 7230 nM T40556 CEA2C7 155531097 Ki = 128 nM T40556 CNB0Z3 155531098 Ki = 0.5 nM T40556 CS48EO 155531154 IC50 = 545.2 nM T40556 CL9VB6 155531262 IC50 = 5000 nM T40556 C84UXT 155531461 IC50 = 3620 nM T40556 CV2DU3 155531469 IC50 = 2400 nM T40556 CJ93LE 155531635 IC50 = 5011.87 nM T40556 CJ3XQ0 155531658 IC50 = 63.1 nM T40556 CPY0W4 155531898 Ki = 65.4 nM T40556 COI6T9 155532041 Ki = 1.1 nM T40556 CME45L 155532169 IC50 = 1584.89 nM T40556 C7IG9L 155532175 IC50 = 47 nM T40556 CQN6G3 155532286 IC50 = 690 nM T40556 CH80JY 155532661 IC50 = 67 nM T40556 C82UPM 155532741 IC50 = 10000 nM T40556 CQ6G3D 155532785 IC50 > 10000 nM T40556 C7LUW5 155533038 IC50 = 71 nM T40556 CE3R7T 155533055 IC50 = 63 nM T40556 CQ63ZW 155533302 IC50 = 9065 nM T40556 C1HOJ8 155533481 Ki = 34.8 nM T40556 C3P5FB 155533716 IC50 = 240 nM T40556 CYL48U 155533835 IC50 = 790 nM T40556 CCS3Z2 155533896 IC50 = 630.96 nM T40556 CSDL12 155533972 Ki = 0.9 nM T40556 CY37NL 155534118 IC50 = 240 nM T40556 CRVW82 155534145 Ki = 83.7 nM T40556 CWQ9I0 155534265 IC50 = 220 nM T40556 CH39ZT 155534291 IC50 = 70 nM T40556 C9A7EM 155534450 Ki = 12.59 nM T40556 CZY5G8 155534471 IC50 = 2250 nM T40556 CFV0X3 155534492 IC50 = 81 nM T40556 CAEQ29 155534550 IC50 = 25118.86 nM T40556 C4Y2JK 155534563 Ki = 249 nM T40556 C0QV9U 155534567 IC50 = 3200 nM T40556 CWP5Z4 155534721 Ki = 0.8 nM T40556 CJUX72 155534784 IC50 = 860 nM T40556 C8R6ZI 155534867 IC50 = 8200 nM T40556 CS57MP 155535054 IC50 = 46 nM T40556 C6OP0S 155535292 Ki = 14.8 nM T40556 CBTQ04 155535301 Ki = 1.1 nM T40556 CY08SU 155535485 IC50 = 31622.78 nM T40556 C91UNV 155535585 IC50 = 2550 nM T40556 CS8XB0 155535800 IC50 = 850 nM T40556 CFM46E 155535834 IC50 = 1810 nM T40556 CG7X4Y 155536037 Ki = 12.59 nM T40556 CTYQ86 155536169 IC50 > 10000 nM T40556 C7L0ZW 155536305 IC50 = 54.8 nM T40556 C0HI7N 155536879 EC50 > 10000 nM T40556 CX01IJ 155536900 IC50 = 665.7 nM T40556 CV1FU3 155537340 IC50 = 7200 nM T40556 C02DSM 155537630 IC50 = 316.23 nM T40556 CS1KL9 155538190 IC50 = 27.5 nM T40556 CZS3A1 155538358 IC50 = 110 nM T40556 CEZJ39 155538579 IC50 = 709.4 nM T40556 C9ISB5 155538742 IC50 > 50118.72 nM T40556 CF3YQ7 155539142 IC50 = 82 nM T40556 C87NOU 155539256 IC50 = 203 nM T40556 C71XPS 155539263 Ki = 918 nM T40556 C1MQP2 155539283 IC50 = 50118.72 nM T40556 C9UP3S 155539471 IC50 = 46 nM T40556 CDCP41 155539526 IC50 = 503.2 nM T40556 C8TSQ0 155539582 IC50 = 4400 nM T40556 C7WY9X 155539828 IC50 = 113 nM T40556 CW1Z8F 155539966 Ki = 109 nM T40556 CE0FM3 155540495 IC50 = 6170 nM T40556 C62EMT 155540785 IC50 = 760 nM T40556 CV1GR7 155540862 Ki = 1.2 nM T40556 CABF92 155541119 IC50 = 750 nM T40556 C7VRN8 155541456 IC50 = 750 nM T40556 C6SG3O 155541524 IC50 = 44 nM T40556 C9SIN5 155541564 IC50 = 107 nM T40556 CXTO91 155541586 IC50 = 31622.78 nM T40556 C4UC2G 155542752 IC50 = 7300 nM T40556 CNSP97 155542781 IC50 > 50118.72 nM T40556 CF95RE 155542833 IC50 > 10000 nM T40556 CJ94RY 155543134 Ki = 17.4 nM T40556 CT8E7F 155543334 Ki = 147 nM T40556 C6FHM8 155543582 IC50 = 31622.78 nM T40556 C0IQ7Y 155544012 IC50 > 10000 nM T40556 CK2N5P 155544158 IC50 = 172.1 nM T40556 CL9Q5B 155545073 IC50 = 20 nM T40556 C2UN1K 155545446 IC50 > 10000 nM T40556 CDQ8J3 155545496 IC50 = 1600 nM T40556 C1Z6RY 155545684 Ki = 0.8 nM T40556 C1JSY3 155545907 IC50 > 10000 nM T40556 CM51BF 155546089 IC50 = 39810.72 nM T40556 CP5VY1 155546607 IC50 = 316.23 nM T40556 CH9Y8A 155546620 IC50 = 328 nM T40556 CFTR89 155546746 IC50 = 39810.72 nM T40556 CK10MI 155546815 IC50 = 48 nM T40556 C71QBN 155546897 IC50 = 550 nM T40556 CAV1O8 155546975 IC50 = 141 nM T40556 C82ZVR 155547161 Ki = 2.9 nM T40556 CUX25H 155547195 Ki = 15.9 nM T40556 CQPY75 155547500 IC50 = 5170 nM T40556 CAI8W4 155547542 IC50 = 29 nM T40556 C8ZGQ3 155547993 Ki = 174 nM T40556 CAI1K4 155548058 IC50 = 95.2 nM T40556 CNW10F 155548254 IC50 = 57 nM T40556 CST0E6 155548743 Ki = 28 nM T40556 CI12GZ 155548897 Ki = 0.5 nM T40556 CQNO46 155548910 IC50 = 31622.78 nM T40556 C8O0PK 155549061 Ki = 74.7 nM T40556 CH62AP 155549078 IC50 = 348.2 nM T40556 C4RO8G 155549970 Ki = 1.1 nM T40556 CBHN73 155550160 IC50 = 20 nM T40556 C6C3KR 155550228 IC50 = 106.7 nM T40556 CTPL52 155550409 IC50 = 540 nM T40556 C3VAJ9 155550685 IC50 = 6710 nM T40556 CNU0K9 155551427 Ki = 68 nM T40556 C1YK4R 155551595 IC50 = 708.7 nM T40556 C2VN6S 155551648 IC50 = 140 nM T40556 CJL84K 155551807 IC50 = 95 nM T40556 C4VKR0 155551851 IC50 > 50118.72 nM T40556 COG5X6 155551883 IC50 = 2410 nM T40556 CE5PB8 155551897 IC50 = 23870 nM T40556 C2FWB9 155551946 IC50 = 39810.72 nM T40556 CJ49KI 155552070 IC50 = 5920 nM T40556 C68TQG 155552169 IC50 = 260.3 nM T40556 CE6XY4 155552472 IC50 = 10 nM T40556 C5Q8NM 155552649 IC50 > 10000 nM T40556 C6SE1C 155552754 Ki = 68 nM T40556 CXB3A0 155552980 IC50 = 16341 nM T40556 C7RPH3 155553336 IC50 < 50 nM T40556 CKA2N6 155553423 Ki = 5.8 nM T40556 CHL5S0 155553610 Ki = 12.3 nM T40556 C1TLD7 155553647 IC50 = 50.12 nM T40556 CT35SU 155553650 IC50 = 39810.72 nM T40556 C4DXG8 155553846 IC50 = 3888 nM T40556 CTRE24 155554039 Ki = 0.8 nM T40556 C0VP2N 155554114 Ki = 66.2 nM T40556 CH8L1V 155554197 IC50 = 3480 nM T40556 CJN29K 155554220 IC50 = 292 nM T40556 C0SYN6 155554629 IC50 = 25118.86 nM T40556 C4UER7 155554809 IC50 = 271.2 nM T40556 CW5LG1 155554980 Ki = 284 nM T40556 CB6Q5S 155555122 IC50 = 2226 nM T40556 C7OR6T 155555165 Ki = 13 nM T40556 C1T5RH 155555385 IC50 = 61 nM T40556 CF2H3O 155555451 IC50 > 10000 nM T40556 CM7FN8 155555499 IC50 = 1170 nM T40556 CDO08V 155555578 IC50 > 50118.72 nM T40556 C12QHG 155555950 IC50 > 50118.72 nM T40556 CP2BX0 155556096 IC50 = 7943.28 nM T40556 C6JSF2 155556169 IC50 = 220 nM T40556 C83KNU 155556217 IC50 = 573.1 nM T40556 CZJ7Y4 155556283 Ki = 1.7 nM T40556 C7S8GF 155556284 IC50 > 50118.72 nM T40556 CFS7H1 155556713 IC50 = 2600 nM T40556 C5CSM3 155556861 IC50 = 1600 nM T40556 C6N1CG 155557122 IC50 > 50118.72 nM T40556 CUQ53E 155557175 IC50 = 150 nM T40556 C57UCJ 155557247 Ki = 2.1 nM T40556 C3BY7N 155557439 IC50 = 4500 nM T40556 CYM3K9 155557522 IC50 = 15848.93 nM T40556 C4I0RK 155557553 IC50 = 18500 nM T40556 C7T1PN 155557578 IC50 = 560 nM T40556 CK8O4T 155557646 IC50 > 50118.72 nM T40556 CE07MN 155557702 Ki = 68.8 nM T40556 CWHA10 155558023 IC50 > 10000 nM T40556 CM23TJ 155558268 Ki = 0.9 nM T40556 C6D4EN 155558707 IC50 = 391.3 nM T40556 C2P3TA 155558894 IC50 = 35.1 nM T40556 CSGH17 155559412 IC50 > 50118.72 nM T40556 CD4ML1 155559481 IC50 = 76 nM T40556 C5S7RE 155559494 IC50 > 10000 nM T40556 CH24ZI 155559572 IC50 = 3600 nM T40556 C2MX6K 155559855 IC50 = 158.49 nM T40556 C1C9VU 155559875 Ki = 41.5 nM T40556 CZ94JU 155560004 IC50 = 217.1 nM T40556 CSF23U 155560126 Ki = 0.6 nM T40556 C5X6EL 155560182 IC50 > 50118.72 nM T40556 CBNS45 155560213 IC50 = 155 nM T40556 C5DLU8 155560288 IC50 = 1320 nM T40556 CS1C5W 155560567 IC50 > 50118.72 nM T40556 CK45IM 155560616 Ki = 4.3 nM T40556 CI91CS 155560656 IC50 = 24000 nM T40556 C3UC7H 155560671 IC50 = 25118.86 nM T40556 C1CHQ8 155560764 Ki = 21.3 nM T40556 CG19QD 155561005 IC50 = 162 nM T40556 CI1ZU8 155561055 IC50 = 9600 nM T40556 CU2O6Z 155561457 Ki = 1.4 nM T40556 CH0Z1P 155561539 IC50 > 10000 nM T40556 CRNC43 155561660 IC50 = 1400 nM T40556 CZA5N1 155561689 EC50 = 9110 nM T40556 C3RYM5 155561853 IC50 = 10041 nM T40556 C7FCQ9 155562154 IC50 = 79000 nM T40556 CM25ZY 155562178 IC50 = 680 nM T40556 C0JQF4 155562547 IC50 = 79.43 nM T40556 C0Y9BU 155562553 IC50 < 100 nM T40556 C2U1DO 155563442 IC50 = 709.1 nM T40556 CI3F7H 155563640 IC50 = 1584.89 nM T40556 CJ1ZK6 155563724 IC50 = 2400 nM T40556 CK0BV2 155564034 IC50 = 2511.89 nM T40556 CGWP21 155564141 IC50 = 889 nM T40556 CQK18D 155564294 IC50 = 4810000 nM T40556 C5NU8A 155564453 IC50 = 1500 nM T40556 C7ICA9 155564455 EC50 > 10000 nM T40556 CJ3ZR5 155564460 IC50 = 220 nM T40556 C47LAU 155564565 IC50 = 14.4 nM T40556 C8LF6O 155564647 IC50 = 2436 nM T40556 C7EDG4 155564694 IC50 = 10000 nM T40556 CC8O2L 155565265 IC50 = 50.12 nM T40556 C68CBM 155565352 IC50 = 25.9 nM T40556 C4VSH5 155565624 IC50 = 810.4 nM T40556 CY83NZ 155565684 Ki = 2.8 nM T40556 C17NSI 155566209 IC50 = 1960 nM T40556 CZC03T 155566251 IC50 = 176 nM T40556 CK9C6J 155566327 IC50 = 334.2 nM T40556 CXRJ70 155566441 IC50 > 50118.72 nM T40556 CJ5B1M 155566905 Ki = 2.1 nM T40556 C2PIK0 155567275 IC50 > 501187.23 nM T40556 CZK10H 155567377 IC50 > 10000 nM T40556 CM5FL1 155567534 IC50 > 50118.72 nM T40556 C8ZS0C 155567638 IC50 = 21 nM T40556 CMV75T 155567768 Ki = 1230 nM T40556 CXZG79 155567978 Ki = 1.8 nM T40556 C7C9DH 155568184 IC50 > 50118.72 nM T40556 CV9L7S 155568572 Ki = 1.3 nM T40556 CUWO65 155568681 IC50 = 68 nM T40556 C06GWZ 155568932 Ki = 24.7 nM T40556 CZ2VN0 155569163 IC50 > 50118.72 nM T40556 C48AYZ 155569378 IC50 = 800 nM T40556 CN56LR 155569534 Ki = 6.31 nM T40556 CNF0G9 155569554 IC50 = 480 nM T40556 D00DXI 135566302 Ki = 10850 nM T40556 D00XRH 91820725 IC50 = 1258.93 nM T40556 D01YSN 57345400 IC50 = 26 nM T40556 D03BTJ 15990224 IC50 = 3162.28 nM T40556 D03LIP 13953710 IC50 = 15.5 nM T40556 D03LNF 71271629 IC50 = 220 nM T40556 D03XXT 72201027 IC50 = 3200 nM T40556 D09HBR 135566899 Ki < 85 nM T40556 D09VHS 3971 IC50 = 9050 nM T40556 D09ZPM 1091852 IC50 = 79432.82 nM T40556 D0C2JS 71291068 IC50 = 92 nM T40556 D0F5TZ 91827383 IC50 = 2511.89 nM T40556 D0H3TC 54669868 IC50 = 4786.3 nM T40556 D0J3JI 90488984 IC50 = 600 nM T40556 D0J6XI 1253361 IC50 = 2500 nM T40556 D0N5BI 91668541 IC50 = 5011.87 nM T40556 D0O2RX 71624782 IC50 = 371.54 nM T40556 D0O6XT 91827373 IC50 = 3700 nM T40556 D0Q7IU 40642506 IC50 = 10400 nM T40556 D0T3WL 73010930 IC50 > 50000 nM T40556 D0T3YY 59190723 Ki = 16.7 nM T40556 D0V8MX 606801 IC50 = 4300 nM T40556 D0VC0I 5169 IC50 = 2500 nM T40556 D0WU1S 52912189 Ki = 9 nM T40556 D0Y3OO 11327430 IC50 = 1000 nM T15700 D0J3SU 9847835 EC50 > 5000 nM T15700 D0U6WQ 153270 IC50 = 40 nM T15700 COW5R3 608841 Ki = 2700 nM T15700 CI0DG1 764318 IC50 > 200000 nM T15700 C5WKA9 2779120 Ki = 30000 nM T15700 C1V6CM 2821593 IC50 = 75000 nM T15700 C7CLA9 2821595 IC50 = 62000 nM T15700 C2U4HS 2821632 IC50 > 200000 nM T15700 CMP1F6 2821634 IC50 > 200000 nM T15700 CR7N4T 2821636 IC50 = 60000 nM T15700 COTB47 2821639 IC50 > 200000 nM T15700 C1JRB7 2821640 IC50 = 60000 nM T15700 C12EXP 2821660 IC50 > 200000 nM T15700 CGOH73 2821679 IC50 > 200000 nM T15700 CPA63I 3107941 IC50 = 76100 nM T15700 C6SO2K 3708081 IC50 > 200000 nM T15700 C1RUH9 4246483 IC50 > 100000 nM T15700 CT4YC1 5287959 IC50 = 3850 nM T15700 C3T8NF 5288850 IC50 > 50000 nM T15700 CO58XD 5311161 IC50 > 100000 nM T15700 C1KR5B 5327301 Ki = 4000 nM T15700 C37TKL 5327302 Ki = 150 nM T15700 C64ZMN 5327304 Ki = 880 nM T15700 C3IZ2W 5327307 Ki = 19000 nM T15700 C16DTL 5327308 Ki = 50 nM T15700 C4O3QY 5327309 Ki = 330 nM T15700 C3GUM7 5327310 Ki = 710 nM T15700 C3LZX9 8027611 IC50 > 50000 nM T15700 CFN2P6 9800285 Ki = 80000 nM T15700 CE7I9W 9806986 IC50 = 1.75 nM T15700 CYFG94 9807028 IC50 = 6600 nM T15700 CD3P2F 9807170 IC50 = 9.57 nM T15700 C3S1EP 9807375 IC50 = 9.1 nM T15700 C13PRZ 9809421 IC50 = 490 nM T15700 CLTO67 9821317 IC50 = 7 nM T15700 C4XO3K 9821545 Ki = 49000 nM T15700 CJI5T3 9823027 IC50 = 7 nM T15700 C74QTI 9823074 IC50 = 770 nM T15700 C6S3KT 9840223 Ki > 25000 nM T15700 CN02PU 9849845 IC50 = 6.42 nM T15700 C5MCX4 9849846 IC50 = 7.56 nM T15700 CDC86G 9850642 IC50 = 1.66 nM T15700 CJO3A5 9851213 IC50 = 2.73 nM T15700 C56LDH 9851279 IC50 = 3290 nM T15700 C6O0QH 9852052 IC50 = 0.016 nM T15700 CD05OL 9867192 IC50 = 179 nM T15700 C2N3LE 9871540 IC50 = 2.26 nM T15700 CX17DM 9871570 IC50 > 10 nM T15700 CF0V7B 9871631 IC50 = 6.59 nM T15700 CLQH78 9892350 IC50 = 7.65 nM T15700 CW75OE 9892652 IC50 = 2.9 nM T15700 C3YAL4 9895375 IC50 = 1500 nM T15700 C2DMG1 9914167 IC50 > 50000 nM T15700 CK15RJ 9916276 IC50 = 8.22 nM T15700 C0D2IJ 9936767 IC50 = 2.09 nM T15700 CG90WC 9939287 IC50 = 810 nM T15700 CFCK64 9939773 IC50 = 6300 nM T15700 CN63JG 9958554 IC50 = 3.3 nM T15700 C9CV0Y 10001828 IC50 = 770 nM T15700 CW4Q3N 10031194 IC50 = 2400 nM T15700 CHWA42 10074552 IC50 = 7800 nM T15700 CZ3IH4 10414828 IC50 = 2000 nM T15700 CX67SZ 10826725 Ki = 31000 nM T15700 CDX7A4 10963183 Ki = 28000 nM T15700 C7HSX0 11189577 IC50 = 336 nM T15700 CM8O6L 11257152 IC50 = 17 nM T15700 CCV6T0 11374367 IC50 = 6 nM T15700 C4F8DC 11444079 IC50 > 500000 nM T15700 CDT9G3 11467504 IC50 = 4.03 nM T15700 CV4CP9 11496333 IC50 > 50000 nM T15700 CGE2J0 11497112 IC50 > 50000 nM T15700 C6IS9K 11509289 IC50 > 50000 nM T15700 C6L2MY 11509300 IC50 > 50000 nM T15700 CC31QO 11509301 IC50 > 50000 nM T15700 CS8OX7 11510566 IC50 > 500000 nM T15700 C7FY9B 11512139 IC50 > 50000 nM T15700 C15VFG 11515586 IC50 > 500000 nM T15700 CW6PC0 11519268 IC50 > 50000 nM T15700 CZC5D9 11525874 IC50 > 50000 nM T15700 C5BNE1 11533326 IC50 > 50000 nM T15700 CDK3Z5 11533935 IC50 > 10000 nM T15700 C4IC7E 11541867 IC50 > 500000 nM T15700 C3USR9 11543714 IC50 = 575 nM T15700 C3P2GZ 11548424 IC50 > 500000 nM T15700 CVX4M6 11548909 EC50 > 5000 nM T15700 C17OJS 11572844 IC50 = 1120 nM T15700 CF0V3P 11576540 IC50 > 50000 nM T15700 C1T9DY 11576622 IC50 > 50000 nM T15700 C03KPR 11576852 EC50 > 5000 nM T15700 CN67DR 11583840 IC50 > 50000 nM T15700 CPD0M8 11584106 IC50 > 50000 nM T15700 CL16IM 11591540 IC50 > 50000 nM T15700 CE2TX6 11591919 IC50 > 500000 nM T15700 CG4Z9A 11598106 IC50 > 10000 nM T15700 CV6MF1 11614728 IC50 > 500000 nM T15700 CFP19E 11619968 IC50 > 50000 nM T15700 CA0LH6 11624920 IC50 > 50000 nM T15700 CEY39D 11628992 IC50 > 500000 nM T15700 C6UAV3 11632008 IC50 = 425 nM T15700 C6Y5MG 11634372 IC50 > 50000 nM T15700 CKJE92 11634649 IC50 > 50000 nM T15700 C4QB6F 11635889 IC50 = 4 nM T15700 C91JNO 11639020 IC50 = 288 nM T15700 C4MCW2 11646889 IC50 = 835 nM T15700 C2KFU3 11647018 IC50 > 50000 nM T15700 CH20JE 11652994 IC50 = 24700 nM T15700 CN32TX 11664423 IC50 > 500000 nM T15700 CUD05C 11670894 IC50 > 50000 nM T15700 CX97NT 11684618 IC50 > 50000 nM T15700 C05YRV 11699954 IC50 > 500000 nM T15700 CKEX64 11700402 IC50 > 500000 nM T15700 C89COT 11705942 IC50 > 50000 nM T15700 C86PAH 11712912 IC50 > 50000 nM T15700 CY90EM 11712953 IC50 = 506 nM T15700 CNV75J 11713799 IC50 > 10000 nM T15700 C7QK5F 11755713 IC50 = 15500 nM T15700 CRWS56 16046172 IC50 = 9400 nM T15700 C7YI1R 16725993 IC50 = 14 nM T15700 CXH9M5 16749067 IC50 > 50000 nM T15700 C2DJ5W 16749068 IC50 > 50000 nM T15700 COM07G 16749069 IC50 > 50000 nM T15700 CPG8Q0 16749161 IC50 > 50000 nM T15700 CG84TK 16749162 IC50 > 50000 nM T15700 CT3HD1 16749163 IC50 > 50000 nM T15700 CZM4X2 16749164 IC50 > 50000 nM T15700 CUZ8N4 16749267 IC50 > 50000 nM T15700 CMEK96 16749268 IC50 > 50000 nM T15700 C01HBN 16749269 IC50 > 50000 nM T15700 CWG3C8 16749270 IC50 > 50000 nM T15700 C8R3GD 16749271 IC50 > 50000 nM T15700 CW9HL5 23645230 IC50 = 1885 nM T15700 C5G2IL 23645238 IC50 = 92 nM T15700 C74OPE 23645239 IC50 = 22050 nM T15700 CK7B2A 23645240 IC50 = 1150 nM T15700 C8YA0T 23645241 IC50 = 3650 nM T15700 C8J7UY 23645242 IC50 = 7270 nM T15700 C3MGC1 23645243 IC50 = 7340 nM T15700 CLSU45 23645244 IC50 = 9175 nM T15700 C95KHP 23645245 IC50 = 8000 nM T15700 C08UYG 23645246 IC50 > 10000 nM T15700 C6YEO7 23645247 IC50 = 9580 nM T15700 CFH23D 23645248 IC50 = 13800 nM T15700 CY0M3Z 23645249 IC50 = 12300 nM T15700 C4TIM0 23645250 IC50 > 10000 nM T15700 CZ9HT6 23645253 IC50 = 2900 nM T15700 CZ59CM 23645306 IC50 = 8700 nM T15700 CNU1R6 23645307 IC50 = 3300 nM T15700 C8WF2G 23645308 IC50 = 14000 nM T15700 CBSA54 23645309 IC50 = 9300 nM T15700 C9ZJ4W 23655167 IC50 = 93000 nM T15700 CTI80F 25178948 EC50 > 5000 nM T15700 C2GI4J 25178949 EC50 > 5000 nM T15700 CQ2GM9 25178950 EC50 > 5000 nM T15700 C4GFV6 25179140 EC50 > 5000 nM T15700 CYL36B 25179141 EC50 > 5000 nM T15700 CGC69Q 25179143 EC50 > 5000 nM T15700 C27YJF 25179144 EC50 > 5000 nM T15700 C2YTB7 25179145 EC50 > 5000 nM T15700 C6GTV3 25179324 EC50 > 5000 nM T15700 CIC46T 25179513 EC50 > 5000 nM T15700 CK96WB 25179514 EC50 > 5000 nM T15700 CGX78D 25217029 IC50 > 50000 nM T15700 CW2L9Q 25217030 IC50 > 50000 nM T15700 C8UTC4 25217031 IC50 > 50000 nM T15700 CZ43KQ 25217032 IC50 > 50000 nM T15700 C2P9NI 25217145 IC50 > 25000 nM T15700 C8C9XU 42618276 IC50 > 50000 nM T15700 CFO93N 42618277 IC50 > 50000 nM T15700 CS1KQ0 42618278 IC50 > 50000 nM T15700 CVI16X 42618279 IC50 > 50000 nM T15700 C3MRA0 42618280 IC50 > 50000 nM T15700 C8UO9S 42618281 IC50 > 50000 nM T15700 C68NPR 42618282 IC50 > 50000 nM T15700 CL41SD 42618283 IC50 > 50000 nM T15700 CJ7U2E 42618284 IC50 > 50000 nM T15700 CZL8C7 42618285 IC50 > 50000 nM T15700 CNIQ28 42618286 IC50 > 50000 nM T15700 C91OMB 42618287 IC50 > 50000 nM T15700 C5AC1L 42618288 IC50 > 50000 nM T15700 CFU5T2 42618289 IC50 > 50000 nM T15700 CK9H3M 42618290 IC50 > 50000 nM T15700 CV4H2J 42618291 IC50 > 50000 nM T15700 C7VPU3 42618292 IC50 > 50000 nM T15700 C6R2FM 42618293 IC50 > 50000 nM T15700 CD8WB9 44304162 Ki > 50000 nM T15700 C9RLK1 44309811 Ki = 350 nM T15700 CAB39E 44331552 IC50 = 4140 nM T15700 CE0FW4 44331565 IC50 = 3040 nM T15700 C8SZN9 44331566 IC50 = 1690 nM T15700 CMFW61 44331567 IC50 = 1450 nM T15700 CHYL38 44331577 IC50 = 15000 nM T15700 C1I9QH 44331578 IC50 = 4720 nM T15700 C4VGZ1 44331579 IC50 = 6050 nM T15700 CRZ01H 44331580 IC50 = 7530 nM T15700 CFOR90 44331674 IC50 = 3860 nM T15700 CK7VI8 44331675 IC50 = 1710 nM T15700 CH7GS4 44331676 IC50 > 10000 nM T15700 C4FOD3 44331693 IC50 > 10000 nM T15700 CJY5L2 44331739 IC50 = 4950 nM T15700 C8N2GQ 44331740 IC50 = 1750 nM T15700 CW9K4Q 44331815 IC50 = 1860 nM T15700 CT76DG 44331816 IC50 = 8600 nM T15700 CC70GF 44331830 IC50 = 8700 nM T15700 CNJ19L 44331876 IC50 = 12700 nM T15700 C46IPA 44331879 IC50 > 10000 nM T15700 CP0Y8M 44331898 IC50 = 80 nM T15700 CF3R6W 44331908 IC50 > 10000 nM T15700 C0S8LV 44331910 IC50 = 30 nM T15700 CTM5W1 44331914 IC50 = 31 nM T15700 C0YZ9O 44331915 IC50 = 12 nM T15700 C4NK1S 44331942 IC50 = 80 nM T15700 CXKY19 44331943 IC50 = 10000 nM T15700 C3FC8D 44331944 IC50 > 10000 nM T15700 CH1ZF2 44331953 IC50 = 990 nM T15700 C0QJ8V 44331957 IC50 = 19590 nM T15700 C1HBX6 44331963 IC50 = 50000 nM T15700 C7UXK5 44331964 IC50 = 11960 nM T15700 C42PGN 44331965 IC50 = 670 nM T15700 C5J7KX 44331966 IC50 > 10000 nM T15700 CG83FS 44331967 IC50 = 2240 nM T15700 CGAJ95 44331977 IC50 = 733 nM T15700 CCYX84 44331980 IC50 = 1200 nM T15700 C5UIO2 44331987 IC50 = 4350 nM T15700 C0PM5C 44332004 IC50 = 12200 nM T15700 C4ENB1 44332005 IC50 = 615 nM T15700 CFK4Z1 44332024 IC50 = 2430 nM T15700 CTM3G2 44332026 IC50 = 16300 nM T15700 C48ZEW 44332028 IC50 > 50000 nM T15700 C30MKG 44332029 IC50 > 50000 nM T15700 C7OS9X 44332050 IC50 = 4340 nM T15700 C9Y6NP 44332051 IC50 = 13400 nM T15700 C0VGF8 44332058 IC50 = 3870 nM T15700 CQU84D 44332068 IC50 = 9280 nM T15700 CBL91D 44332078 IC50 = 5900 nM T15700 C4VCM3 44332093 IC50 = 15200 nM T15700 C92QVT 44332108 IC50 = 7420 nM T15700 CQLZ09 44332109 IC50 = 29100 nM T15700 C4CUL6 44332112 IC50 = 1420 nM T15700 CN2YM6 44332113 IC50 = 200 nM T15700 C4CY8K 44332118 IC50 = 450 nM T15700 CXZ2N1 44332120 IC50 = 3640 nM T15700 CD56PK 44332121 IC50 = 4020 nM T15700 C5A6OJ 44332128 IC50 > 50000 nM T15700 C6IZ2R 44332129 IC50 = 11000 nM T15700 C5DY0G 44332136 IC50 = 48 nM T15700 CQ1K9H 44332311 IC50 = 7.6 nM T15700 C9LOS2 44332330 IC50 = 9810 nM T15700 C2U6GB 44332331 IC50 = 5230 nM T15700 CH01QW 44332332 IC50 = 11200 nM T15700 C8D5TB 44364680 Ki = 810 nM T15700 C1ZHJ7 44384620 EC50 = 25000000 nM T15700 CA74KZ 44386296 EC50 = 4000000 nM T15700 CV23MO 44389236 IC50 > 10 nM T15700 C2I3VJ 44389240 IC50 = 0.22 nM T15700 CI89LR 44389245 IC50 > 10 nM T15700 CR7VM8 44389295 IC50 = 4.92 nM T15700 CU5VW3 44389297 IC50 = 9.26 nM T15700 C5P8TU 44389299 IC50 > 10 nM T15700 C5YC0O 44389306 IC50 = 6.22 nM T15700 C1FMX8 44389307 IC50 > 10 nM T15700 CB6US3 44389310 IC50 > 10 nM T15700 CC8S0I 44389315 IC50 = 2.46 nM T15700 CEO19T 44389316 IC50 > 10 nM T15700 CRC82Z 44389318 IC50 = 9.92 nM T15700 CPE0S2 44389319 IC50 > 10 nM T15700 CC8MG3 44389324 IC50 = 0.49 nM T15700 C9X1RJ 44389325 IC50 = 0.99 nM T15700 CF0CN3 44389326 IC50 > 10 nM T15700 C7LQP0 44389331 IC50 = 9.22 nM T15700 CEQ2L1 44389335 IC50 > 10 nM T15700 C9C3JB 44389337 IC50 > 10 nM T15700 CU0I3N 44389338 IC50 = 7.38 nM T15700 CALT41 44389340 IC50 = 10 nM T15700 C5LO3T 44389347 IC50 = 4.29 nM T15700 CJA5K7 44389348 IC50 = 6.02 nM T15700 C2WS9G 44389351 IC50 = 5.28 nM T15700 CEH8Z5 44389369 IC50 > 10 nM T15700 CBJ15U 44389458 IC50 > 10 nM T15700 C2OU7Z 44389483 IC50 > 10 nM T15700 CA81WI 44389513 IC50 = 9.54 nM T15700 CL4G2Y 44389531 IC50 = 9.04 nM T15700 CX5Y3A 44389532 IC50 = 6.48 nM T15700 CEH02Q 44389544 IC50 > 10 nM T15700 CXN03I 44389545 IC50 = 5.95 nM T15700 CQPY50 44391346 IC50 = 1625 nM T15700 CJQE23 44391364 IC50 = 5380 nM T15700 CE3YN5 44391369 IC50 = 1320 nM T15700 CWVF04 44391384 IC50 = 4505 nM T15700 C0J6SU 44391388 IC50 = 5830 nM T15700 C24KOF 44391455 IC50 > 10000 nM T15700 CA58XR 44391530 IC50 = 975 nM T15700 CU3ZB5 44391569 IC50 = 104 nM T15700 CI7F3G 44391602 IC50 = 635 nM T15700 CL73OE 44391603 IC50 = 280 nM T15700 CIU0P1 44391632 IC50 = 98 nM T15700 C5J4LV 44403257 IC50 > 10000 nM T15700 CYNX83 44403316 IC50 > 10000 nM T15700 CAGR97 44403319 IC50 > 10000 nM T15700 CWQ21I 44403320 IC50 > 10000 nM T15700 C5P9KT 44403321 IC50 > 10000 nM T15700 CB2E3T 44403325 IC50 > 10000 nM T15700 CAU6G0 44404870 IC50 = 1823 nM T15700 CU4N7M 44404871 IC50 = 4811 nM T15700 C3RL0N 44404877 IC50 = 7540 nM T15700 CGQ1U4 44404931 IC50 = 10000 nM T15700 CKU1S0 44404937 IC50 = 3046 nM T15700 CO38AJ 44405528 IC50 = 384 nM T15700 CBY58A 44405529 IC50 = 247 nM T15700 CVJ8Z3 44405532 IC50 = 481 nM T15700 CHG69W 44405540 IC50 = 911 nM T15700 CZ8Y2S 44405566 IC50 = 264 nM T15700 C6X1JT 44405629 IC50 = 13 nM T15700 CK62FC 44405634 IC50 = 160 nM T15700 COXU97 44405637 IC50 = 917 nM T15700 CGV2B4 44405663 IC50 = 429 nM T15700 CFX81S 44405672 IC50 = 38 nM T15700 CS40LN 44405689 IC50 = 50 nM T15700 C2MOF9 44405695 IC50 = 5 nM T15700 CYG86L 44405707 IC50 = 384 nM T15700 CMUS37 44405733 IC50 = 106 nM T15700 CJ07FL 44405737 IC50 = 601 nM T15700 C1VY3T 44405740 IC50 = 595 nM T15700 C0DL8M 44405752 IC50 = 283 nM T15700 CB7V6W 44405784 IC50 = 1585 nM T15700 C1VW8E 44405799 IC50 = 3770 nM T15700 CH6CN5 44405800 IC50 = 670 nM T15700 C8EK9W 44405805 IC50 = 4190 nM T15700 CWP51F 44405816 IC50 = 6450 nM T15700 CEY48X 44405818 IC50 = 7900 nM T15700 CXA87L 44405820 IC50 = 1600 nM T15700 CM2GJ1 44405827 IC50 = 448 nM T15700 CAY57C 44405829 IC50 = 1550 nM T15700 C7LEI3 44405837 IC50 = 2590 nM T15700 CUY3M1 44414212 IC50 = 2100 nM T15700 C79OFE 44414311 IC50 >= 10000 nM T15700 CFL7O1 44414418 IC50 = 4300 nM T15700 C2DIQ3 44414439 IC50 = 130 nM T15700 C9Q4KR 44414440 IC50 = 6300 nM T15700 C0FQ1E 44414442 IC50 = 3900 nM T15700 C50NAG 44414456 IC50 = 1170 nM T15700 C34DMY 44414457 IC50 = 1200 nM T15700 CV0EW7 44414458 IC50 = 70 nM T15700 CL29BC 44414459 IC50 = 2600 nM T15700 CV96AO 44414484 IC50 = 230 nM T15700 C9P7ZA 44414485 IC50 = 300 nM T15700 C4GWP5 44414501 IC50 = 3120 nM T15700 CY0VU1 44414502 IC50 = 420 nM T15700 C8H5YL 44414541 IC50 = 2200 nM T15700 CW45EL 44414543 IC50 = 90 nM T15700 CB0M5Q 44414572 IC50 = 310 nM T15700 CXEH76 44414573 IC50 = 3200 nM T15700 CMI4Z9 44414574 IC50 = 1800 nM T15700 CJT30G 44414592 IC50 = 2700 nM T15700 CIQ36K 44414642 IC50 >= 10000 nM T15700 CW0MH5 44416221 IC50 > 10000 nM T15700 COS6D2 44416249 IC50 = 8500 nM T15700 CL6YM3 44416250 IC50 = 5000 nM T15700 CL8IC5 44416262 IC50 > 10000 nM T15700 C21FST 44416320 IC50 = 5200 nM T15700 C3FO6V 44416321 IC50 > 10000 nM T15700 CN91HB 44416330 IC50 = 9500 nM T15700 CF6J2T 44416331 IC50 = 7000 nM T15700 CJ6QG4 44417479 IC50 > 500000 nM T15700 C7RX9I 44418960 Ki = 540 nM T15700 C0YBP2 44428506 IC50 = 2935 nM T15700 CY3K9C 44428508 IC50 = 2160 nM T15700 CF2NM3 44428511 IC50 = 1451 nM T15700 CD9VU2 44428513 IC50 = 4196 nM T15700 CT8R6X 44428515 IC50 = 1231 nM T15700 CS87UF 44428517 IC50 = 1957 nM T15700 C12AHI 44428519 IC50 = 1184 nM T15700 CWG6S2 44428521 IC50 = 554 nM T15700 CYHS50 44428523 IC50 = 162 nM T15700 CERS10 44428524 IC50 = 537 nM T15700 C2Q0FD 44428525 IC50 = 2688 nM T15700 C9R5MT 44428526 IC50 = 2110 nM T15700 C3CY9O 44428527 IC50 = 1606 nM T15700 CM50ES 44428528 IC50 = 10000 nM T15700 CP3XJ0 44428530 IC50 = 109 nM T15700 C62JNP 44428532 IC50 = 1085 nM T15700 C5AE0W 44428534 IC50 = 887 nM T15700 CE0V2J 44428536 IC50 = 448 nM T15700 CL6K0W 44428539 IC50 = 471 nM T15700 CXR1V5 44434249 IC50 = 6 nM T15700 C31JIN 44438441 IC50 > 10000 nM T15700 CKI30F 44438442 IC50 = 300 nM T15700 CNO1C0 44438443 IC50 = 3050 nM T15700 CI1G7O 44438444 IC50 = 1000 nM T15700 C5Y1IC 45379628 IC50 = 100000 nM T15700 C3DRB6 45496892 IC50 > 200000 nM T15700 CDY2W5 49796910 IC50 = 2.1 nM T15700 C0HMT1 49797331 IC50 = 163.5 nM T15700 C3M2BW 52918163 IC50 > 50000 nM T15700 CF24IM 52918177 IC50 > 50000 nM T15700 CR9I7F 52918178 IC50 > 50000 nM T15700 C2VPU1 52918179 IC50 > 50000 nM T15700 C8Z2TQ 54580470 IC50 > 50000 nM T15700 CMU0B4 54581481 IC50 > 50000 nM T15700 CCS8Y3 54581987 IC50 > 50000 nM T15700 CJEP38 54582484 IC50 > 50000 nM T15700 C61NWL 54582924 IC50 > 50000 nM T15700 CO0AG3 54583923 IC50 > 25000 nM T15700 CI2DL4 54583924 IC50 > 50000 nM T15700 CV2WU1 54583925 IC50 > 50000 nM T15700 CXA51D 54584867 IC50 > 50000 nM T15700 C8YSL0 54585834 IC50 > 50000 nM T15700 C9B5OF 54586343 IC50 > 50000 nM T15700 C7A8ER 54587376 IC50 > 50000 nM T15700 CGY3W2 71471109 IC50 = 2620 nM T15700 CANH70 71716242 IC50 = 4100 nM T15700 C40WIR 71718085 IC50 = 5930 nM T15700 CU75VK 71719897 IC50 = 600 nM T15700 CBV6F1 71720507 IC50 = 12900 nM T15700 CXZ6D5 73347105 EC50 = 25000000 nM T15700 C4U5TO 76311196 IC50 > 10000 nM T15700 CSI53E 76311200 IC50 > 10000 nM T15700 CNOL37 76311201 IC50 > 10000 nM T15700 C8IS5Q 76314800 IC50 > 10000 nM T15700 CK41QI 76314804 IC50 > 10000 nM T15700 CHS61N 76314805 IC50 > 10000 nM T15700 CDY7K0 76318413 IC50 > 10000 nM T15700 CB2N6G 76322078 IC50 > 10000 nM T15700 C8SPW6 76322082 IC50 > 10000 nM T15700 CC2EP6 76325698 IC50 > 10000 nM T15700 CFY79U 76332916 IC50 > 10000 nM T15700 CD35SI 76332917 IC50 > 10000 nM T15700 C3FQX0 76336535 IC50 > 10000 nM T15700 CV4PE6 76336536 IC50 > 10000 nM T15700 CQ9H4U 86277844 IC50 = 6800 nM T15700 CKCI60 90663142 IC50 = 17 nM T15700 C9QKI3 127020966 IC50 > 100000 nM T15700 CV04JO 127037715 IC50 > 50000 nM T15700 CJ27CG 127042051 IC50 > 50000 nM T15700 CAT46D 127042341 IC50 > 50000 nM T15700 CWM2E8 133081971 IC50 > 9999 nM T15700 CU42CE 155567829 IC50 > 100000 nM T15700 D0L9AX 644345 IC50 = 130 nM T15700 D0N5MU 4117381 Ki > 50000 nM T15700 D0N8TA 11466200 IC50 = 4.2 nM T15700 D0Q9XX 515950 Ki > 50000 nM T15700 D0V6DX 10640 IC50 = 1910 nM T15700 D0Y5IQ 44255320 IC50 = 5000 nM T44818 D05EJG 6305 Ki = 11500000 nM T44818 D06MHZ 66558287 IC50 < 1000 nM T44818 D0DP5I 121328278 IC50 > 10000 nM T44818 D0J1HB 23063810 IC50 > 10000 nM T44818 D0PM5U 135564890 IC50 = 242 nM T44818 D0WR7B 122650373 IC50 = 47 nM T44818 C9SC4E 46702 EC50 = 950 nM T44818 C9E7UR 79703 EC50 > 25000 nM T44818 CR36LZ 235240 Ki = 16000 nM T44818 CFPL09 236715 IC50 = 52900 nM T44818 CA1H8B 336270 IC50 = 733 nM T44818 CL2JH7 336699 IC50 = 71010 nM T44818 C46VHU 478572 IC50 = 53 nM T44818 C72ZLN 478574 IC50 = 68 nM T44818 CC7IW3 478577 IC50 = 215 nM T44818 C2ZR8M 478643 IC50 = 59 nM T44818 CY38AJ 478645 IC50 = 241 nM T44818 CZT01E 478647 Ki = 8410 nM T44818 CXYV26 849731 IC50 = 711 nM T44818 C47XAO 849732 IC50 = 6460 nM T44818 CB27WS 849733 IC50 = 561 nM T44818 C5S9DF 849734 IC50 = 1745 nM T44818 C34QEU 849735 IC50 = 1088 nM T44818 CSC0B6 1041635 IC50 = 7380 nM T44818 CF3XV1 1382046 EC50 = 9700 nM T44818 CB2K7L 2747165 IC50 > 25000 nM T44818 C5T3HX 2748785 EC50 = 85 nM T44818 C6KJL8 2750134 EC50 > 25000 nM T44818 CE6H2V 2759980 EC50 > 25000 nM T44818 CU27GW 2806085 EC50 = 820 nM T44818 C12IDC 3901929 IC50 = 46810 nM T44818 CV10YZ 4190125 IC50 = 53380 nM T44818 CNUQ02 4456830 IC50 = 38310 nM T44818 CL82TX 6400901 IC50 > 100000 nM T44818 CGP9S8 6409664 IC50 > 100000 nM T44818 C3AV5I 6419227 IC50 > 100000 nM T44818 CAVT12 9812842 IC50 > 100000 nM T44818 C4UYP5 9815283 IC50 > 100000 nM T44818 C4QZ1I 9877471 IC50 > 100000 nM T44818 C7N9PW 9877511 IC50 > 100000 nM T44818 C6NS2U 9899225 IC50 > 100000 nM T44818 CU3RN8 9920462 IC50 > 100000 nM T44818 C69CDF 9920916 IC50 > 100000 nM T44818 C2PCN3 9964175 IC50 > 100000 nM T44818 CUP4N1 9964258 IC50 > 100000 nM T44818 C2UQ5N 10014426 Ki = 30 nM T44818 C4RKW2 11255489 IC50 = 3000 nM T44818 C32WXK 11275256 IC50 > 100000 nM T44818 CZS6U0 11694196 IC50 > 100000 nM T44818 CIFV43 12760724 EC50 > 25000 nM T44818 CQJP83 12949094 IC50 > 25000 nM T44818 C39AWQ 13393248 IC50 = 60220 nM T44818 CYE1A6 14171304 IC50 = 1600 nM T44818 CUD51F 16740669 EC50 = 1400 nM T44818 CS84LJ 19702149 IC50 > 100000 nM T44818 C08CBI 21723626 IC50 > 100000 nM T44818 CGM9O7 22009901 IC50 > 100000 nM T44818 CBSK32 22424949 EC50 = 210 nM T44818 C1BI5L 22989786 IC50 = 5150 nM T44818 C0Z3PM 24741909 IC50 = 58330 nM T44818 CQJ8F1 25211983 IC50 = 3350 nM T44818 C0ZJY1 25211984 IC50 = 7150 nM T44818 CRG7J1 28806364 Ki = 32400 nM T44818 C3HLB4 45117984 EC50 > 25000 nM T44818 CE5JF9 45790362 EC50 = 250 nM T44818 CEQ2B0 53391619 IC50 = 10000 nM T44818 CF6X2A 53391627 IC50 = 5000 nM T44818 C42UIZ 53391725 Ki = 21000 nM T44818 CA19IT 57611775 IC50 = 27200 nM T44818 CPG21M 58911926 IC50 = 270 nM T44818 CVJ0N6 60154724 IC50 > 100000 nM T44818 CA1TW8 60154725 IC50 > 100000 nM T44818 CA8W4D 60154726 IC50 > 100000 nM T44818 CW0FS2 60156091 IC50 > 100000 nM T44818 CDM64W 60156092 IC50 > 100000 nM T44818 CS31CB 60156093 IC50 > 100000 nM T44818 C2LSA3 60156094 IC50 > 100000 nM T44818 CA34YM 60156095 IC50 > 100000 nM T44818 C0JI9X 61393224 EC50 = 1500 nM T44818 CZM31Y 62502228 IC50 = 29 nM T44818 CHX38T 66558199 IC50 = 20 nM T44818 C8CMD0 70874604 EC50 = 250 nM T44818 CJ24YM 70914178 IC50 < 1000 nM T44818 C2TC8W 70914230 EC50 = 2000 nM T44818 CNUF17 71458329 IC50 > 100000 nM T44818 CJ0UW8 82366003 EC50 = 1500 nM T44818 C4W8RF 82410733 IC50 > 25000 nM T44818 CGT4O9 85469240 Ki = 170 nM T44818 C8T0MJ 85469241 Ki = 1560 nM T44818 C5SWD9 85469242 IC50 = 270 nM T44818 CA5CG1 85469243 IC50 = 290 nM T44818 C5R6WS 85469292 IC50 = 470 nM T44818 C3Z8YX 91758737 Ki = 310 nM T44818 C7FA1J 105422590 EC50 = 360 nM T44818 CL7KP4 118895094 IC50 = 190 nM T44818 CM46PT 121254880 IC50 = 60 nM T44818 CSF24O 122193552 IC50 = 768 nM T44818 C25XGV 122193553 IC50 = 1586 nM T44818 CV30GB 122193590 IC50 = 167 nM T44818 C4RSB3 122193591 IC50 = 312 nM T44818 C4N9HG 122193592 IC50 = 90 nM T44818 C8A0DL 122193593 IC50 = 181 nM T44818 CR27QH 122193594 IC50 = 59 nM T44818 CXY02W 122193595 IC50 = 48 nM T44818 CJ6RO8 122193596 IC50 = 30 nM T44818 CL7S4T 122193597 IC50 = 176 nM T44818 CCL63T 122193598 IC50 = 116 nM T44818 CP93QC 122193599 IC50 = 30 nM T44818 CIDM29 122193600 IC50 = 209 nM T44818 C2U6VA 122193601 IC50 = 145 nM T44818 CC6VJ5 122525709 IC50 = 180 nM T44818 CY0X9D 122525711 IC50 = 60 nM T44818 CZE79W 122525712 Ki = 120 nM T44818 C7K5BJ 122529269 IC50 = 309 nM T44818 C98MWA 122529271 IC50 = 71 nM T44818 CH28KJ 122529388 IC50 = 43 nM T44818 CX9JY7 122529428 IC50 = 58 nM T44818 CF4D7J 122529456 IC50 = 26 nM T44818 C34WLE 122551145 IC50 = 27 nM T44818 C51WNS 122606362 IC50 = 70 nM T44818 CGO29F 122608329 IC50 = 70 nM T44818 CXS30F 122650362 IC50 > 10000 nM T44818 CU2K4P 122650372 IC50 = 132 nM T44818 C3RCU4 122650378 IC50 = 215 nM T44818 C3LY8T 122650476 IC50 = 394 nM T44818 CP9EY1 122650500 IC50 = 371 nM T44818 CN6MK9 122650505 IC50 = 338 nM T44818 CHZY51 122650508 IC50 = 639 nM T44818 CS47AD 122650581 IC50 = 65 nM T44818 C3YM4T 124927661 IC50 = 1200 nM T44818 CY7G4D 129282405 EC50 = 50 nM T44818 CQ97RT 129282436 EC50 = 36 nM T44818 CL9J8N 129282617 EC50 = 70 nM T44818 CP09TF 129282671 EC50 = 210 nM T44818 C42ZDX 129282689 EC50 = 72 nM T44818 C3GA7K 129282703 EC50 = 130 nM T44818 CV28YE 129282706 EC50 = 65 nM T44818 C7LG2X 129282851 EC50 = 1400 nM T44818 C3SGN0 129282870 EC50 = 50 nM T44818 CU70NI 129282903 EC50 = 7400 nM T44818 C3CH6E 129283030 EC50 = 380 nM T44818 C7FXS8 129283166 EC50 = 39 nM T44818 C32WDC 129283174 EC50 = 32 nM T44818 C9HZ2S 129283211 EC50 = 54 nM T44818 C5L7MR 129283737 EC50 = 87 nM T44818 CE19JM 129296385 EC50 = 48 nM T44818 C56BAE 129296459 EC50 = 3000 nM T44818 CC47DZ 134132888 IC50 = 3000 nM T44818 C8QOD7 134138847 IC50 = 3000 nM T44818 CVB51Y 134141021 IC50 = 3000 nM T44818 CQD8V6 134142830 IC50 = 3000 nM T44818 CV5XQ0 134143523 IC50 = 3000 nM T44818 C2HJ8Z 134146158 IC50 = 3000 nM T44818 C8D9KR 134146460 IC50 = 3000 nM T44818 CSUE71 134149657 IC50 = 3000 nM T44818 CI69YJ 134150572 IC50 = 3000 nM T44818 CM62BZ 134154095 IC50 = 3000 nM T44818 C15WLQ 134154247 IC50 = 3000 nM T44818 C9ZEJ4 134462563 IC50 = 85 nM T44818 CCJ85U 135412567 IC50 = 46240 nM T44818 CB9Q2N 135424953 IC50 = 3000 nM T44818 CXE5S3 135482065 IC50 > 100000 nM T44818 CASN86 135743630 IC50 = 398 nM T44818 C9KHP8 135981331 IC50 > 100000 nM T44818 C1ARX6 137297350 IC50 > 10000 nM T44818 CJ73IG 137390209 EC50 = 33 nM T44818 CD29IP 139507088 IC50 > 10000 nM T44818 CL2AV8 142619909 IC50 = 84000 nM T44818 CM8P4F 142619919 IC50 = 54400 nM T44818 C38SQV 145950032 IC50 = 18000 nM T44818 C3E5BK 145952508 IC50 = 28 nM T44818 C0RGQ7 145952699 EC50 = 77 nM T44818 C6K3PQ 145953664 IC50 > 25000 nM T44818 CW9I0R 145954143 EC50 = 230 nM T44818 CM2Z3H 145957538 EC50 = 18000 nM T44818 C2QC1G 145957647 EC50 > 25000 nM T44818 CBN73E 145971997 EC50 = 340 nM T44818 C71ARM 145972688 EC50 = 810 nM T44818 C8CXN2 145979858 IC50 = 83470 nM T44818 C3UG5E 145980172 IC50 = 684.3 nM T44818 C1IGW2 145980819 IC50 > 100000 nM T44818 CW8B6A 145981750 IC50 = 321.5 nM T44818 CV1RQ9 145981894 IC50 = 39920 nM T44818 CHN2M6 145982993 IC50 > 100000 nM T44818 CCLP04 145983079 IC50 = 1200 nM T44818 C4AKU1 145983122 IC50 > 100000 nM T44818 CPR1W2 145983299 IC50 = 41600 nM T44818 CH1X5E 145984494 IC50 = 7300 nM T44818 CJC34M 145984936 IC50 > 100000 nM T44818 CF3ME9 145985603 IC50 > 100000 nM T44818 CP09AH 145985633 IC50 > 100000 nM T44818 CEJR90 145986692 IC50 > 100000 nM T44818 CJ3TE7 145986756 IC50 = 73.1 nM T44818 C05UPF 145987627 IC50 = 214.5 nM T44818 CGT41S 145987994 IC50 = 54690 nM T44818 CH8S9C 145988339 IC50 > 100000 nM T44818 CB15WE 145990300 IC50 > 100000 nM T44818 CB0ZR4 145992186 IC50 > 100000 nM T44818 CD4WA8 145994224 IC50 = 56120 nM T44818 C8J3TV 146669430 IC50 = 2940 nM T44818 C36ISR 153434865 IC50 > 10000 nM T44818 C3IH8C 155510739 IC50 = 20 nM T44818 C4JB1R 155511259 IC50 = 183 nM T44818 CLWA53 155511337 IC50 = 1029 nM T44818 C7PTI6 155511361 IC50 = 48800 nM T44818 CWDH25 155511770 IC50 = 3320 nM T44818 CAG5F0 155513388 IC50 = 19100 nM T44818 CHP5L0 155514083 IC50 = 29800 nM T44818 CYFW59 155514258 IC50 = 4530 nM T44818 C3CD4X 155514316 IC50 = 77400 nM T44818 CES90B 155515098 IC50 = 586 nM T44818 CZGI76 155515235 IC50 = 17000 nM T44818 CCJ14L 155516448 IC50 = 114 nM T44818 CJ0FH7 155516689 IC50 = 58700 nM T44818 CH4B9K 155517551 EC50 <= 32 nM T44818 CJA45U 155518566 IC50 = 3920 nM T44818 C2F6OX 155520170 IC50 = 5000 nM T44818 C3ZP5H 155521897 IC50 = 22500 nM T44818 CLY12I 155525014 IC50 = 49700 nM T44818 CIO1A3 155532842 EC50 = 71 nM T44818 C70XJB 155533149 IC50 = 2770000 nM T44818 CG1K4V 155533289 IC50 = 4540 nM T44818 C4H8XB 155536067 IC50 = 2540 nM T44818 C0O4AQ 155536365 IC50 = 5700 nM T44818 C0HXA8 155538715 IC50 = 95 nM T44818 CFKI70 155539267 IC50 = 3960 nM T44818 CD3Y5U 155540952 IC50 = 7150 nM T44818 C4C6RX 155541201 IC50 = 579 nM T44818 CF3AW0 155541799 IC50 = 12000 nM T44818 C02NAK 155542721 IC50 = 226 nM T44818 CNPU01 155546283 IC50 = 374 nM T44818 CH96DK 155550037 IC50 = 21800 nM T44818 C2GSR8 155550907 IC50 = 189 nM T44818 C6JV3E 155551216 EC50 = 60 nM T44818 CE95UF 155552938 IC50 = 4410 nM T44818 C8M1QG 155553198 IC50 = 6210 nM T44818 C0ASJ7 155553201 EC50 = 35 nM T44818 CQ6D7M 155555581 IC50 = 195 nM T44818 CO7P3Z 155557740 IC50 = 5620 nM T44818 C4RWF1 155558731 IC50 = 376 nM T44818 C1TIH7 155558824 IC50 = 353 nM T44818 CBYL12 155559016 IC50 = 4000 nM T44818 C25KBO 155562131 IC50 = 3480 nM T44818 C3NDJ2 155562711 IC50 = 9020 nM T44818 CSQ8U0 155562797 IC50 = 793 nM T44818 C4MBN1 155564503 IC50 = 7000 nM T44818 CG02FV 155564613 IC50 = 4820 nM T44818 C5Z8YM 155565919 IC50 = 500 nM T44818 C61SEH 155567075 IC50 = 6370 nM T44818 C07ASO 155567542 IC50 = 1275 nM T44818 CO58ME 155567694 EC50 = 130 nM T44818 C2O8RC 155568012 IC50 = 123000 nM T44818 CSB45Q 155569293 EC50 = 62 nM T44818 CC8LV5 155569500 IC50 > 25000 nM T44818 D01HST 1085108 IC50 > 62500 nM T44818 D0I9AT 73549 IC50 = 140 nM T44818 D0O3IE 137153 IC50 > 100000 nM T44818 D0Z3NE 478573 IC50 = 40 nM T91397 D0E3TC 44259 IC50 = 1040 nM T91397 CACS26 11561968 Ki = 1500 nM T91397 CU0E8O 11690457 Ki = 160 nM T91397 CB0AP2 11705863 Ki = 660 nM T91397 COH62U 60097413 IC50 > 4000 nM T91397 C1MR8Q 60097495 IC50 > 10000 nM T91397 D0J3LR 11634725 Ki > 10000 nM T46465 D0W9JM 60927 Ki = 1000 nM T46465 D04ZIJ 5478883 IC50 = 0.42 nM T46465 D0X8AU 446837 IC50 = 30 nM T46465 C2V3YA 90664069 Ki = 110 nM T46465 CAD6F5 44330836 Ki = 110 nM T46465 C3G6QJ 24051 IC50 = 1000 nM T46465 CZ0JE7 31222 IC50 = 1000 nM T46465 C9ZTV0 77079 IC50 = 1000 nM T46465 CGN71C 213804 IC50 = 5000 nM T46465 CYJ72V 226139 IC50 = 1000 nM T46465 COA7U4 330448 IC50 = 24000 nM T46465 C2OS0K 407573 IC50 = 19000 nM T46465 C6HBV9 444581 IC50 = 2880 nM T46465 C2AX7O 445304 Ki = 85 nM T46465 C6AP4F 446918 Ki = 100 nM T46465 CQC83A 475853 Ki = 3800 nM T46465 C53JAZ 669278 IC50 = 24000 nM T46465 CSQ2I1 877648 IC50 = 24000 nM T46465 C1W5JF 895406 IC50 = 24000 nM T46465 C3DA6G 1134093 Ki = 4600 nM T46465 CY0L8J 1742906 Ki = 2000 nM T46465 CJF8Q3 1743728 IC50 = 8990 nM T46465 C13SGI 1829851 IC50 = 7000 nM T46465 CB8OL5 2818163 IC50 = 9470 nM T46465 C2G0QD 2835079 Ki = 7000 nM T46465 CMEV06 2860116 IC50 = 24000 nM T46465 CR7K6L 2971411 IC50 = 24000 nM T46465 CVR7P3 3781218 IC50 = 1000 nM T46465 CG2W7Q 3832424 Ki = 1600 nM T46465 CGZ6F5 4685845 Ki = 50 nM T46465 CXE8N9 5338725 IC50 = 24000 nM T46465 C5ND0S 6520996 Ki = 4000 nM T46465 CPS5Z7 6539218 Ki = 0.56 nM T46465 CV5K3I 6539219 Ki = 46 nM T46465 C7UR8H 6539220 Ki = 11 nM T46465 CYA9X5 6539221 Ki = 0.5 nM T46465 CY6M5W 6539222 Ki = 30 nM T46465 CEX3D8 6539224 Ki = 248 nM T46465 C9DOI1 6539225 Ki = 29 nM T46465 CR7A3L 6539226 Ki = 74 nM T46465 C0H5ZW 6539227 Ki = 25 nM T46465 CUQ6T5 6539228 Ki = 256 nM T46465 C32QNI 6539229 Ki = 68 nM T46465 CZN02I 6539230 Ki = 15 nM T46465 CXPO09 6539231 Ki = 91 nM T46465 C4GX1T 6539232 Ki = 10 nM T46465 C2YKM3 6539233 Ki = 139 nM T46465 COLZ28 6539234 Ki = 284 nM T46465 CJ14EB 6539235 Ki = 348 nM T46465 CQ5O9H 6539236 Ki = 131 nM T46465 CIY71M 6539237 Ki = 144 nM T46465 CIWC50 6539238 Ki = 390 nM T46465 C9VQZ4 6539239 Ki = 230 nM T46465 CT6C2N 6539240 Ki = 4100 nM T46465 C4AXO5 6539241 Ki = 96 nM T46465 CY8HL5 6539242 Ki > 2500 nM T46465 CA78BY 6539243 Ki = 47 nM T46465 CB2O4C 6539244 Ki = 29 nM T46465 CEX54J 6539245 Ki = 59 nM T46465 C61TOP 6539246 Ki = 129 nM T46465 C01MAJ 6539247 Ki = 6 nM T46465 CV7NB4 6539248 Ki = 13 nM T46465 CMHE43 6539249 Ki = 14 nM T46465 CQO6I0 6539250 Ki = 15 nM T46465 CHC57F 6539251 Ki = 181 nM T46465 CT30RS 6539252 Ki = 15 nM T46465 CNZ8E9 6539253 Ki = 8.9 nM T46465 CV9Q8Z 6539254 Ki = 41 nM T46465 C3VB5A 6539255 Ki = 130 nM T46465 C6H5IQ 6539256 Ki = 37 nM T46465 CF30BP 6539257 Ki = 11 nM T46465 CZ40TI 6539258 Ki > 2000 nM T46465 CQLC81 6539259 Ki = 50 nM T46465 CMNF51 6539260 Ki = 4.3 nM T46465 C3WI4Y 6539261 Ki > 2000 nM T46465 CE51XA 6539262 Ki ~ 3300 nM T46465 CN6OX1 6539263 Ki > 2000 nM T46465 CB89QP 6539264 Ki ~ 3200 nM T46465 CB14ZY 6539265 Ki ~ 3500 nM T46465 CBF54P 6539266 Ki = 540 nM T46465 CM6X7H 6539267 Ki = 117 nM T46465 C6RQ9Z 6539268 Ki = 121 nM T46465 C0Y9GC 6539269 Ki = 150 nM T46465 CWIJ07 6539270 Ki = 379 nM T46465 CSD6R5 6539271 Ki = 1430 nM T46465 CWR7C9 6539272 Ki > 2000 nM T46465 CXT20F 6539273 Ki = 930 nM T46465 CURY46 6539274 Ki = 579 nM T46465 CLE4I2 6539275 Ki = 129 nM T46465 C1SUG3 6539276 Ki = 1900 nM T46465 CV2JK1 6539277 Ki = 928 nM T46465 C4HAV1 7514787 IC50 = 6000 nM T46465 C26ZFH 9630864 Ki = 8000 nM T46465 CA46BZ 9633226 Ki = 1200 nM T46465 CKP0I3 9830952 Ki = 3 nM T46465 C7Z8UC 9831520 Ki = 220 nM T46465 CV7J8R 9893943 IC50 = 101 nM T46465 C0HM2T 9895330 Ki = 2 nM T46465 CF7D2T 9960476 Ki = 2 nM T46465 CF18OZ 9961626 Ki = 300 nM T46465 CCTU14 10030581 IC50 = 100 nM T46465 CO7A2D 10033021 Ki = 4.8 nM T46465 C5Y1NI 10120764 IC50 = 511 nM T46465 CZ40NB 10145154 IC50 = 33 nM T46465 C37QPJ 10184491 IC50 = 1700 nM T46465 C18XBZ 10187123 IC50 = 1800 nM T46465 CC6S7R 10229401 IC50 = 13 nM T46465 C1GJK8 10279305 IC50 = 143 nM T46465 CEVR93 10280148 IC50 = 1700 nM T46465 CV8FY1 10302032 IC50 = 70 nM T46465 CKPL79 10302679 IC50 = 104 nM T46465 CT3WY2 10302959 IC50 = 35 nM T46465 C9Z2BY 10327349 Ki = 9 nM T46465 C7AQS8 10348528 IC50 < 100 nM T46465 CJ05CH 10369893 IC50 < 100 nM T46465 C5C0JY 10393370 Ki > 30000 nM T46465 C16FLQ 10407914 IC50 > 1000 nM T46465 C5C8FP 10437723 IC50 = 2000 nM T46465 CL27YN 10462501 Ki = 4.1 nM T46465 C21ANW 10485108 IC50 ~ 40000 nM T46465 CKXB12 10508444 Ki = 4 nM T46465 CPX74Q 10662259 IC50 = 6000 nM T46465 CV01KW 11106059 IC50 = 1000 nM T46465 CR6W3Y 11168223 IC50 = 212 nM T46465 C0J2NU 11204230 Ki = 308 nM T46465 C1YFZ0 11214849 IC50 = 113 nM T46465 CEDP95 11215989 Ki = 55 nM T46465 CENB36 11227366 Ki = 45 nM T46465 C06RKV 11237615 IC50 = 380 nM T46465 CE1B6S 11239445 Ki = 19 nM T46465 CX30NP 11249866 Ki = 214 nM T46465 CZ4X0A 11250844 Ki = 48 nM T46465 C8PHK2 11273154 Ki = 16 nM T46465 C5ZDP8 11284770 IC50 = 145 nM T46465 C2C4XA 11285489 Ki = 0.9 nM T46465 C4BHV0 11285517 Ki = 1.9 nM T46465 C98FEY 11285691 Ki > 5000 nM T46465 C5BO7P 11296167 Ki = 13 nM T46465 C2QK0E 11308017 Ki = 693 nM T46465 C7ER8J 11376724 IC50 = 183 nM T46465 CP2YI7 11387548 IC50 = 463 nM T46465 C1RG5P 11399816 Ki = 4.4 nM T46465 C6UT8Z 11399839 Ki = 1.1 nM T46465 CSJD04 11410402 Ki = 260 nM T46465 CBQO36 11444127 IC50 = 100 nM T46465 C9YKP7 11505733 Ki = 3400 nM T46465 CJ9NL1 11505900 Ki > 5000 nM T46465 C1VEC2 11513333 Ki = 6 nM T46465 C8P5JQ 11513415 Ki = 586 nM T46465 CF2JU9 11520423 Ki = 2100 nM T46465 C6U9JR 11527693 Ki = 168 nM T46465 CKU80T 11534178 Ki > 5000 nM T46465 CKY5C8 11534582 Ki > 5000 nM T46465 CS0H9X 11534953 Ki = 2900 nM T46465 C02DGS 11541427 Ki = 161 nM T46465 C8SFN6 11541810 Ki > 5000 nM T46465 CB59KM 11564069 Ki = 145 nM T46465 C8RPH4 11607313 Ki = 7 nM T46465 C7XU9H 11614671 Ki = 1300 nM T46465 CSR87I 11629093 Ki = 2300 nM T46465 CN9AO7 11636216 Ki = 14 nM T46465 CA45GE 11657449 Ki = 359 nM T46465 CHXL54 11664893 Ki = 10 nM T46465 CM46HF 11671674 IC50 = 31 nM T46465 CXN6V9 11685086 Ki > 5000 nM T46465 CWTA90 11707562 Ki = 142 nM T46465 CIDF31 11721953 Ki = 11 nM T46465 CH1Y8K 11764107 Ki = 1.1 nM T46465 CIN27G 11785613 IC50 = 531 nM T46465 CD1N7A 11787369 Ki = 5.7 nM T46465 C4FZ1S 11838794 IC50 = 6450 nM T46465 C5GK1F 16094654 Ki = 1.9 nM T46465 COIH49 16121203 Ki = 26.3 nM T46465 COU36Z 16645724 IC50 = 24000 nM T46465 C1YE6J 16721109 IC50 = 1816 nM T46465 C50CQN 25066229 IC50 = 4 nM T46465 C4ZQ7Y 28064358 IC50 = 24000 nM T46465 C9H3IT 35756036 IC50 = 10000 nM T46465 C7E0VB 44024156 IC50 = 37700 nM T46465 CD0BS4 44024183 IC50 = 21200 nM T46465 C70PTI 44314034 Ki = 15000 nM T46465 CU9QX3 44314035 Ki = 12000 nM T46465 C80PUQ 44314036 Ki = 5800 nM T46465 C7R6LH 44314039 Ki = 50 nM T46465 CK18PR 44314180 Ki = 410 nM T46465 CPY54X 44314225 Ki = 600 nM T46465 C2KA5V 44314256 Ki = 90 nM T46465 COX2F9 44314257 Ki = 110 nM T46465 CM8EQ3 44314285 Ki = 560 nM T46465 CP2TM3 44314353 Ki = 5600 nM T46465 CMW07C 44314384 Ki = 180 nM T46465 CILR20 44327511 Ki = 180 nM T46465 CQ0F2W 44327556 Ki = 50 nM T46465 CVAJ58 44327796 Ki = 90 nM T46465 C26ZNS 44327901 Ki > 30000 nM T46465 CGJ9B1 44327927 Ki = 410 nM T46465 C8JQ3R 44328032 Ki = 560 nM T46465 CUNS68 44328035 Ki = 220 nM T46465 C3Q0UM 44328055 Ki = 500 nM T46465 CKF62V 44328096 Ki = 12000 nM T46465 CVXC94 44328097 Ki = 5800 nM T46465 C9PCO5 44328098 Ki = 5600 nM T46465 CQGI84 44328099 Ki = 600 nM T46465 CW9CZ3 44328100 Ki = 590 nM T46465 CDV52N 44330684 IC50 = 123 nM T46465 C6X7IR 44335546 Ki = 357 nM T46465 CPL8E9 44338421 IC50 ~ 65000 nM T46465 CHKG96 44338599 IC50 ~ 100000 nM T46465 CM8DR0 44338623 Ki = 490 nM T46465 CY91SZ 44341490 Ki = 41 nM T46465 CAC2O4 44342217 IC50 = 1500 nM T46465 C0HF9G 44418735 Ki = 12.1 nM T46465 CE7TW9 44418736 Ki = 11.2 nM T46465 C2LIW7 44418737 Ki = 103 nM T46465 C6OI8E 44418738 Ki = 9.9 nM T46465 C93HCD 44418739 Ki = 11 nM T46465 CW1NU7 44418740 Ki = 10.6 nM T46465 CF6PJ1 44418741 Ki = 3.9 nM T46465 CY6U5Q 44418742 Ki = 403 nM T46465 CDVZ83 44420384 IC50 = 429 nM T46465 CDC6G4 44420385 IC50 = 589 nM T46465 C1Z9EB 44420386 IC50 = 289 nM T46465 C4OLK1 44420387 IC50 = 6 nM T46465 C5MN2J 44420388 IC50 = 190 nM T46465 C0Z3YP 44420389 IC50 = 165 nM T46465 C8BZ4J 44420390 IC50 = 334 nM T46465 CI2R4O 44420391 IC50 = 531 nM T46465 COJF81 44420392 IC50 = 2345 nM T46465 CY7PQ2 44420393 IC50 = 224 nM T46465 C6PY0U 44420394 IC50 = 439 nM T46465 CB4A9F 44420395 IC50 = 46 nM T46465 C3VF7U 44420396 IC50 = 56 nM T46465 CQ9K2P 44420397 IC50 = 72 nM T46465 C7ZTK3 44420398 IC50 = 74 nM T46465 C1F6YE 44420399 IC50 = 77 nM T46465 CNLR48 44420400 IC50 = 91 nM T46465 C24DUN 44420401 IC50 = 154 nM T46465 CMOI58 44420405 IC50 = 1519 nM T46465 CXTH94 44420406 IC50 = 437 nM T46465 CT28MJ 44420407 IC50 = 574 nM T46465 CXW4H1 44420409 IC50 = 1501 nM T46465 CU76QY 44420410 IC50 = 1912 nM T46465 CLH45S 44420413 IC50 = 334 nM T46465 C1N5TX 44420414 IC50 = 736 nM T46465 CDN15Q 44420415 IC50 = 3015 nM T46465 CU2CD9 44420420 IC50 = 2897 nM T46465 CYTE14 44420421 IC50 = 587 nM T46465 C73WDL 44420424 IC50 = 5266 nM T46465 CB2Q1U 44420429 IC50 = 240 nM T46465 C4XYT1 44420430 IC50 = 642 nM T46465 C03WEN 44420433 IC50 = 670 nM T46465 C0Z1AX 44420434 IC50 = 4553 nM T46465 CL90JP 44420438 IC50 = 464 nM T46465 CB2P3D 44420439 IC50 = 2229 nM T46465 C6JIZ4 44420443 IC50 = 202 nM T46465 CAK03E 44420444 IC50 = 8530 nM T46465 CYN68X 44420449 IC50 = 243 nM T46465 CKZR58 44420450 IC50 = 1491 nM T46465 CA37RB 44420455 IC50 = 369 nM T46465 CJD23P 44420459 IC50 = 200 nM T46465 C5BO7R 44420460 IC50 = 646 nM T46465 C8BL9X 44420461 IC50 = 374 nM T46465 CRH82U 44420462 IC50 = 188 nM T46465 C3PUF9 44420465 IC50 = 3600 nM T46465 CK8QX1 44420466 IC50 = 2549 nM T46465 CRB09U 44425661 Ki = 5 nM T46465 C83ACB 44425670 Ki <= 0.1 nM T46465 C2VE8L 44425675 Ki <= 0.1 nM T46465 CX85GF 44425681 Ki <= 0.1 nM T46465 C8T6YF 44449299 IC50 = 0.13 nM T46465 C7AFS5 44527662 IC50 = 150 nM T46465 CI81AL 44530662 IC50 = 12 nM T46465 CM0A8K 44532986 IC50 = 2700 nM T46465 C0GR5A 44596194 Ki = 830 nM T46465 C3OL5Q 44596195 Ki = 1400 nM T46465 C6R5FM 45267680 IC50 = 590 nM T46465 C1DJR4 45268544 IC50 = 135000 nM T46465 C1UN6X 45268565 IC50 > 25000 nM T46465 C86LOA 45268566 IC50 = 3908 nM T46465 CBA06Z 45268568 IC50 = 11773 nM T46465 C5XUR1 45269412 IC50 = 396000 nM T46465 CC36LM 45269413 IC50 = 9600 nM T46465 CKF16D 45271072 IC50 > 25000 nM T46465 C0Y6CZ 45272777 IC50 = 1510 nM T46465 C8GB5K 45272786 IC50 > 25000 nM T46465 CT6W4D 45273746 IC50 = 12657 nM T46465 CFY29M 45482524 Ki = 7400 nM T46465 CBC9V5 45482525 Ki > 20000 nM T46465 C7AF2S 45482526 Ki > 20000 nM T46465 CT0C5B 45482527 Ki = 440 nM T46465 CX89VL 45482528 Ki = 7600 nM T46465 CXJU16 45482529 Ki = 1700 nM T46465 C14OFW 45482530 Ki > 20000 nM T46465 CA4IM2 46236672 IC50 = 28 nM T46465 C23TKX 46236812 IC50 = 141 nM T46465 CLX98O 46236813 IC50 = 333 nM T46465 CIZD19 46236814 IC50 = 22 nM T46465 CRM4B8 49863568 Ki = 0.4 nM T46465 C0KFO8 53827778 Ki = 50 nM T46465 CZ14SE 54583580 Ki = 10600 nM T46465 C4DF7I 56657884 IC50 = 9.6 nM T46465 CSKW41 56668272 IC50 = 1.51 nM T46465 CJXK94 56671739 IC50 = 0.59 nM T46465 CO3DK2 56671740 IC50 = 135 nM T46465 CO8J5U 56681803 IC50 = 396 nM T46465 C7K3BV 56950381 IC50 = 14700 nM T46465 C0D8IE 57393022 IC50 = 20400 nM T46465 CO8JG5 57393023 IC50 = 48000 nM T46465 C28QVA 57398293 IC50 = 19600 nM T46465 CO2FV3 57398294 IC50 = 30600 nM T46465 CNV5E0 57398295 IC50 = 30500 nM T46465 C71GLZ 57401740 IC50 = 10000 nM T46465 C80LNE 57403473 IC50 = 34000 nM T46465 C3X0EZ 59688843 IC50 = 47 nM T46465 CM9FX0 59688861 IC50 = 67 nM T46465 C0GN4Y 69301328 IC50 < 10 nM T46465 C43UAP 69302432 IC50 < 10 nM T46465 C1OR4B 69783785 IC50 = 10 nM T46465 CI76LZ 69783872 IC50 = 10 nM T46465 CZE7M4 69812537 IC50 = 100 nM T46465 CAME28 69812987 IC50 = 100 nM T46465 CY5A3D 69813189 IC50 = 10 nM T46465 CQJ93U 69813506 IC50 = 10 nM T46465 CV1T6I 69813943 IC50 = 10 nM T46465 CX09SV 69815055 IC50 = 100 nM T46465 C5W9EM 70682473 Ki = 2.3 nM T46465 C1Y4QJ 70682474 Ki = 2.6 nM T46465 CDJ15O 70690877 Ki = 3.8 nM T46465 CGJ3R5 70690878 Ki = 1.3 nM T46465 C5DTE9 71520763 IC50 = 1700 nM T46465 CX34PN 73017594 IC50 = 130 nM T46465 CH5VX9 77722082 IC50 = 10 nM T46465 CUH15E 85343311 IC50 = 4000 nM T46465 CWY76I 85382937 IC50 = 24000 nM T46465 CUW0V3 85384269 IC50 = 3000 nM T46465 CWO38R 85407403 IC50 = 79000 nM T46465 C1BY0I 85470144 IC50 = 570 nM T46465 CSM4C1 86288475 IC50 = 70 nM T46465 CV51KR 86288476 IC50 = 72 nM T46465 C2LJ3N 90654363 Ki = 5.5 nM T46465 C8B7GA 90654364 Ki = 11 nM T46465 C8FN4R 90654365 Ki = 22 nM T46465 C5E3ZF 90654366 Ki = 4.4 nM T46465 C70LGA 90654367 Ki = 4.8 nM T46465 C51FYQ 90654368 Ki = 1.7 nM T46465 CQ9CL3 90654369 Ki = 1.2 nM T46465 CX5H8T 90654370 Ki = 2.3 nM T46465 C6CG8Q 90654371 Ki = 1.1 nM T46465 C7CIE6 90654372 Ki = 1 nM T46465 CAL1E0 90654373 Ki = 5.7 nM T46465 CGS2V7 90654374 Ki = 4.3 nM T46465 CS7ZM6 90655842 IC50 = 270 nM T46465 CQK42C 90655843 IC50 = 190 nM T46465 C64ASN 90655844 IC50 = 150 nM T46465 C65BUL 90655845 IC50 = 600 nM T46465 COG5V7 90655846 IC50 = 500 nM T46465 CL81MW 90655847 IC50 = 500 nM T46465 CAC0H4 90655848 IC50 = 4400 nM T46465 CYS25V 90655849 IC50 = 36 nM T46465 CH9VJ1 90655850 IC50 = 120 nM T46465 CYV70Z 90655851 IC50 = 14000 nM T46465 CPGK89 90655852 IC50 = 320 nM T46465 C48HVL 90655853 IC50 = 24000 nM T46465 C4FR5P 90655854 IC50 = 100 nM T46465 C2GR6X 90655855 IC50 = 110 nM T46465 CL07NM 90655856 IC50 = 800 nM T46465 CXAP16 90655857 IC50 = 190 nM T46465 CY19SM 90664068 Ki = 58.9 nM T46465 C02GTW 102160610 IC50 = 7000 nM T46465 CZK0L7 105539825 IC50 = 340 nM T46465 C2XHZ8 127026505 IC50 = 2300 nM T46465 CB3X2O 127026506 IC50 = 2900 nM T46465 C3DIN6 127027428 IC50 = 1600 nM T46465 CJM2K9 127027429 IC50 = 2500 nM T46465 C9RKY8 127027430 IC50 = 5300 nM T46465 C5XU8O 127027434 IC50 = 230 nM T46465 C51ONW 127027435 IC50 = 150 nM T46465 CZ0M8K 127027436 IC50 = 2000 nM T46465 CR36NE 127027761 IC50 = 2600 nM T46465 CHBD07 127027762 IC50 = 2400 nM T46465 C7ZI6Q 127028384 IC50 = 10700 nM T46465 C7W8FM 127028385 IC50 = 400 nM T46465 C2E3QR 127028386 IC50 = 600 nM T46465 C9H3QY 127028711 IC50 = 2000 nM T46465 C5CR4Z 127028712 IC50 = 10000 nM T46465 CLGB70 127038526 IC50 = 12500 nM T46465 CAT8G7 127039677 IC50 = 32000 nM T46465 C9LAO0 127040014 IC50 = 12000 nM T46465 C0C1AV 127041014 IC50 = 24000 nM T46465 C7AGR0 135474338 IC50 = 53000 nM T46465 C7NI3V 136219158 IC50 = 4620 nM T46465 CR9O7T 145962944 Ki = 1920 nM T46465 CSC48Q 145968177 IC50 = 80 nM T46465 C24PUM 145968574 IC50 = 900 nM T46465 CJ2V6B 145968904 IC50 = 820 nM T46465 C8DOU5 145968976 IC50 = 400 nM T46465 C1D6MG 145969118 IC50 = 75 nM T46465 CT1V0I 145969327 IC50 = 480 nM T46465 CYH45E 145970255 IC50 = 1000 nM T46465 CVAW24 145970337 IC50 = 22 nM T46465 CT57RL 145970338 IC50 = 88 nM T46465 CDR2G9 145970368 IC50 = 93 nM T46465 CM8X7O 145970397 IC50 = 280 nM T46465 CP8A0Z 145970407 IC50 = 23 nM T46465 C4F6NT 145970582 IC50 = 500 nM T46465 CH9P3X 145970804 IC50 = 330 nM T46465 CZ3X4R 145970818 IC50 = 700 nM T46465 CS64YI 145970835 IC50 = 27 nM T46465 C95VSG 145987742 IC50 = 600 nM T46465 C5PA1C 145988827 IC50 = 500 nM T46465 CD4TV5 155510399 IC50 = 350 nM T46465 CRD8I0 155510888 IC50 > 10000 nM T46465 C8XOC6 155511155 IC50 = 2000 nM T46465 C25PLQ 155512213 IC50 = 190 nM T46465 C4JV6P 155515747 IC50 <= 45 nM T46465 CH72PJ 155517364 IC50 = 35 nM T46465 CGV85K 155519272 IC50 > 200000 nM T46465 CLNW30 155519292 IC50 > 20000 nM T46465 C2S4ZM 155519404 IC50 = 2000 nM T46465 CQS70X 155520377 IC50 = 15600 nM T46465 CW89FM 155520640 IC50 = 1100 nM T46465 C85GWP 155521302 IC50 = 270 nM T46465 CAGO28 155523111 IC50 > 10000 nM T46465 COG6S8 155524310 IC50 = 2200 nM T46465 CRVH41 155524341 IC50 = 30 nM T46465 CT3E6C 155524549 IC50 = 380 nM T46465 CMC1B0 155525975 IC50 = 170 nM T46465 C52KOY 155526373 IC50 = 5200 nM T46465 C12KCJ 155527733 IC50 = 1816 nM T46465 C1P9WC 155528474 IC50 = 2700 nM T46465 CTKF74 155530540 IC50 = 7100 nM T46465 CLRB46 155531662 IC50 = 7000 nM T46465 CW0HJ6 155533026 Ki = 50 nM T46465 COI29R 155533689 Ki = 50 nM T46465 CZF54V 155535649 IC50 = 680 nM T46465 CHD2A6 155535700 Ki = 50 nM T46465 CL53AK 155537567 IC50 > 10000 nM T46465 CRN6V8 155537831 IC50 = 160 nM T46465 CO0DJ4 155538305 Ki = 50 nM T46465 CF6E1H 155539416 IC50 > 10000 nM T46465 C03KZX 155539456 IC50 = 850 nM T46465 CVBR73 155539645 IC50 = 5400 nM T46465 CCY83Q 155540092 IC50 = 110 nM T46465 CJB9K1 155540162 IC50 = 39 nM T46465 CFW15C 155540816 IC50 > 10000 nM T46465 C4SP3K 155541193 Ki = 50 nM T46465 CHQD90 155541280 IC50 = 550 nM T46465 C25CXT 155542250 IC50 = 10400 nM T46465 CL9Z6H 155543895 IC50 > 10000 nM T46465 C14SPW 155548636 IC50 > 10000 nM T46465 CIY4E8 155550401 Ki = 50 nM T46465 CAQ1C3 155551571 Ki = 50 nM T46465 CSC98L 155554367 IC50 = 10 nM T46465 C9HX4E 155555414 IC50 = 150 nM T46465 C2B8TR 155556406 IC50 = 1000 nM T46465 C9HK3D 155556455 IC50 = 1950 nM T46465 CMN6E1 155556535 IC50 = 500 nM T46465 C7DH9B 155556912 IC50 = 107 nM T46465 CVQ7G3 155559904 IC50 = 600 nM T46465 C86SOP 155561681 IC50 = 9000 nM T46465 C9DW8H 155563121 IC50 = 10 nM T46465 C5JRM8 155564950 IC50 = 70 nM T46465 CYPV36 155565800 IC50 = 8 nM T46465 CK1U0Y 155566830 IC50 = 50 nM T46465 C1XE0F 155566846 IC50 = 600 nM T46465 C9R2GU 155567898 IC50 = 4190 nM T46465 D00QMZ 44314223 Ki = 220 nM T46465 D00ZMK 49862502 Ki = 1.2 nM T46465 D01RIP 44588309 Ki = 14 nM T46465 D01TFQ 44588301 Ki = 9 nM T46465 D02BVS 49862500 Ki = 17 nM T46465 D02CKL 44588300 Ki = 132 nM T46465 D03BZY 44425663 Ki = 5 nM T46465 D03TFP 49862507 Ki = 4.2 nM T46465 D04QEO 44425662 Ki = 18 nM T46465 D04QUO 25147780 Ki = 21 nM T46465 D04RUS 44588310 Ki = 39 nM T46465 D05DNU 44588315 Ki = 23 nM T46465 D05GIB 16122614 Ki = 3 nM T46465 D05HFQ 44425672 Ki = 4 nM T46465 D05KWN 49862498 Ki = 6.5 nM T46465 D05XTX 44588306 Ki = 55 nM T46465 D06EJX 25147781 Ki = 10 nM T46465 D06MPP 44588296 Ki = 479 nM T46465 D06MZB 44588293 Ki = 55 nM T46465 D06NEW 44588299 Ki = 10 nM T46465 D06QBK 49862499 Ki = 9.1 nM T46465 D07NFJ 44314383 Ki = 220 nM T46465 D08AES 11578664 Ki = 1500 nM T46465 D08FQX 44588320 Ki = 21 nM T46465 D08IXO 44425659 Ki = 0.2 nM T46465 D08SCG 44327926 Ki = 440 nM T46465 D08XLM 44314315 Ki = 500 nM T46465 D09DNT 44425655 Ki = 15 nM T46465 D09XFQ 44588302 Ki = 10 nM T46465 D0A5AT 44588291 Ki = 145 nM T46465 D0D5GN 44425676 Ki = 9 nM T46465 D0E6JX 44588305 Ki = 28 nM T46465 D0E7XR 44588316 Ki = 25 nM T46465 D0F8OH 44588311 Ki = 782 nM T46465 D0G0JA 44588307 Ki = 38 nM T46465 D0G1AF 44588314 Ki = 5 nM T46465 D0G6SP 44588317 Ki = 7 nM T46465 D0H1ZT 44588298 Ki = 10 nM T46465 D0H6LQ 44588313 Ki = 19 nM T46465 D0H6UX 49862501 Ki = 8.5 nM T46465 D0IM5H 44588319 Ki = 26 nM T46465 D0J4NN 49862506 Ki = 0.1 nM T46465 D0JI2X 44314268 Ki = 590 nM T46465 D0JV0F 44588303 Ki = 126 nM T46465 D0K4WS 44588312 Ki = 23 nM T46465 D0M4JP 49862508 Ki = 10 nM T46465 D0M9UG 44425667 Ki = 12 nM T46465 D0N9ON 44588294 Ki = 153 nM T46465 D0O0EA 44588304 Ki = 29 nM T46465 D0O2YF 44425680 Ki = 4 nM T46465 D0O8JQ 44588308 Ki = 25 nM T46465 D0P1MT 49862503 Ki = 0.1 nM T46465 D0PW4M 49862504 Ki = 0.68 nM T46465 D0Q9EB 65012 Ki = 36 nM T46465 D0R0ZC 44588318 Ki = 30 nM T46465 D0S3BO 9895503 Ki = 0.5 nM T46465 D0S4BV 657149 IC50 = 34 nM T46465 D0T3KK 44588295 Ki = 4 nM T46465 D0UX4C 44425679 Ki = 17 nM T46465 D0V2ER 44588292 Ki = 42 nM T46465 D0X2CX 44425657 Ki = 9 nM T46465 D0XU6H 44425666 Ki = 4 nM T46465 D0Y1VG 44588297 Ki = 112 nM T46465 D0YL4X 44425671 Ki = 16 nM T46465 D0Z3GC 49862505 Ki = 5.1 nM T46465 D0Z5MR 44588321 Ki = 6 nM T17523 D07UHS 107970 EC50 = 0.3 nM T17523 D07FKQ 44599207 EC50 = 750 nM T17523 D07UGA 5283560 IC50 = 1.04 nM T17523 D0I2RB 11502996 Ki = 28.8 nM T17523 D0L9KH 44623998 EC50 = 147 nM T17523 D0K4BI 10223146 IC50 > 1000 nM T17523 D0PW0R 71547555 IC50 > 10000 nM T17523 CXSD93 878124 IC50 = 497 nM T17523 C3RZ6P 904918 EC50 > 10000 nM T17523 C1SXH9 1114196 IC50 = 165 nM T17523 C5ODX0 1363299 IC50 = 2000 nM T17523 C7QC0W 1776080 EC50 = 205 nM T17523 CPO6B9 2740144 IC50 > 10000 nM T17523 C7N5UR 4107292 IC50 > 10000 nM T17523 CBPA36 4469648 IC50 = 41 nM T17523 CIA43B 4492589 IC50 = 78 nM T17523 CW8P0C 4780551 EC50 = 162 nM T17523 C89ATE 5309153 EC50 > 50000 nM T17523 C72DNW 9796603 IC50 = 2500 nM T17523 C7FGR9 9979368 IC50 = 40 nM T17523 CI3K9Z 10023913 EC50 = 450 nM T17523 CZLT30 10045980 IC50 = 70 nM T17523 CA4HX3 10125861 IC50 = 76 nM T17523 C8KXE2 10125862 IC50 = 1200 nM T17523 CG6O1W 10125882 IC50 = 600 nM T17523 CN8H2S 10127475 IC50 = 1600 nM T17523 CCG97S 10127776 IC50 = 80 nM T17523 CO06YT 10150171 IC50 = 1.7 nM T17523 CE9WX6 10172338 IC50 = 240 nM T17523 CSV6Q3 10174181 IC50 = 33 nM T17523 C5XFN7 10174255 IC50 = 10000 nM T17523 CG3DX8 10193676 IC50 = 4000 nM T17523 C5HJB9 10195325 IC50 = 790 nM T17523 CY1T7W 10215138 IC50 = 140 nM T17523 CN2FJ9 10216035 IC50 > 10000 nM T17523 C6NP8S 10217498 IC50 = 1300 nM T17523 C9KH2F 10236683 IC50 > 10000 nM T17523 CN93ZD 10249887 IC50 = 370 nM T17523 C6H9VI 10249979 IC50 = 370 nM T17523 C2O4UR 10251062 IC50 = 240 nM T17523 C2YZC3 10271422 IC50 = 210 nM T17523 CN0EC2 10286857 IC50 = 590 nM T17523 C5MDF6 10288527 IC50 = 1500 nM T17523 CJ26CW 10308738 IC50 = 1400 nM T17523 C2U3LT 10309022 IC50 > 10000 nM T17523 CPK61C 10310952 IC50 = 2800 nM T17523 C3SM5Z 10317453 IC50 = 150 nM T17523 CG89DO 10363915 IC50 = 75 nM T17523 CDV3W7 10384596 IC50 = 16 nM T17523 C8WL6R 10408874 IC50 = 49 nM T17523 COQ65E 10409838 IC50 > 10000 nM T17523 CI3EW1 10430549 IC50 = 70 nM T17523 CAL72D 10476387 IC50 = 90 nM T17523 C9NRD6 11168252 IC50 = 340 nM T17523 CZ3T0G 11177439 EC50 = 10 nM T17523 CD8T1W 11222939 EC50 = 0.7 nM T17523 CUR1P8 11224984 EC50 = 1108 nM T17523 CFPH94 11248292 IC50 = 2700 nM T17523 CK65MP 11271470 IC50 > 10000 nM T17523 CYH0U8 11408903 IC50 = 120 nM T17523 CER35T 11466640 IC50 = 2400 nM T17523 CW51YT 11495139 IC50 = 150 nM T17523 CDE78J 11496072 IC50 > 10000 nM T17523 C7EOU1 11501764 IC50 > 1000 nM T17523 CR1ME9 11501873 EC50 > 10000 nM T17523 CS27OX 11502026 IC50 = 4300 nM T17523 CL50IH 11503967 IC50 = 13.1 nM T17523 CAG0Y9 11540052 IC50 = 4.17 nM T17523 CVW6Q3 11575787 IC50 = 89 nM T17523 CB75ZP 11575913 EC50 > 10000 nM T17523 CXS54Q 11603220 IC50 > 1000 nM T17523 CCW90K 11603726 EC50 > 10000 nM T17523 C96LNP 11604577 IC50 = 68 nM T17523 CAN4Q9 11611053 EC50 > 10000 nM T17523 C41XAE 11624780 EC50 > 10000 nM T17523 CCY7J2 11626664 EC50 > 10000 nM T17523 CA8W5N 11646599 EC50 > 10000 nM T17523 CYS5F1 11653967 IC50 = 520 nM T17523 CMJ32O 11662328 IC50 > 10000 nM T17523 C8CQ2N 11675907 EC50 = 91 nM T17523 C3Q9JR 11682677 EC50 = 150 nM T17523 CVG41H 11682696 EC50 > 10000 nM T17523 CQRA36 11683935 IC50 = 6.15 nM T17523 CCF80W 11689680 EC50 > 10000 nM T17523 C8XLO4 11690779 IC50 = 123 nM T17523 C0BR1U 11696807 IC50 = 640 nM T17523 CK5S1L 11697013 EC50 > 10000 nM T17523 C4G2OP 11743459 IC50 = 430 nM T17523 CZ6YN9 11752659 IC50 = 640 nM T17523 CLHA36 11869937 EC50 > 10000 nM T17523 C03OUS 11977938 EC50 = 58 nM T17523 CDI32A 16038017 EC50 > 10000 nM T17523 CGAD08 17253208 EC50 > 50000 nM T17523 CIEK03 17253281 EC50 > 50000 nM T17523 C6HB9A 21455530 IC50 = 800 nM T17523 C6I0ED 24812110 IC50 = 15 nM T17523 C0O9UG 24825338 EC50 > 10000 nM T17523 CB82GW 24825339 IC50 > 10000 nM T17523 C1TGE9 25008420 IC50 = 4.4 nM T17523 C14EAK 25110484 EC50 > 50000 nM T17523 C01FRW 25110488 EC50 > 50000 nM T17523 CXU68J 25110496 EC50 > 50000 nM T17523 CI2VH9 25110498 EC50 > 50000 nM T17523 CLEF36 25110499 EC50 > 50000 nM T17523 C10HKX 25192001 EC50 = 5.39 nM T17523 CXVJ06 33291425 EC50 = 232 nM T17523 C48TPJ 42630194 EC50 = 239 nM T17523 CDL1C8 44125170 EC50 > 41686.94 nM T17523 CG73ST 44138103 EC50 > 100000 nM T17523 CH8CM7 44341291 IC50 = 880 nM T17523 CQR2G1 44341399 IC50 = 140 nM T17523 C95GIJ 44342175 EC50 = 120 nM T17523 C7YT1J 44342219 EC50 = 880 nM T17523 CLXY90 44342331 EC50 = 1400 nM T17523 CI01UD 44342339 EC50 = 1500 nM T17523 CAUQ90 44342468 EC50 = 910 nM T17523 CMKZ19 44344194 IC50 = 200 nM T17523 CLQ25X 44344210 IC50 = 650 nM T17523 C1SP9M 44344338 IC50 > 10000 nM T17523 C2D5LZ 44344360 IC50 = 900 nM T17523 CT4NW0 44344390 IC50 = 140 nM T17523 C9S2FH 44344404 IC50 = 230 nM T17523 CY9C1D 44344412 IC50 = 840 nM T17523 CLDU29 44344413 IC50 = 24 nM T17523 C91OKY 44344446 IC50 = 1400 nM T17523 CL3CT8 44344456 IC50 = 94 nM T17523 C5KA6D 44394117 IC50 > 10000 nM T17523 CU7L0K 44394153 IC50 = 920 nM T17523 CT8UN6 44394161 IC50 > 10000 nM T17523 C9E6CF 44394169 IC50 = 870 nM T17523 C8H0XM 44394191 IC50 = 8.4 nM T17523 CH2A5S 44394211 IC50 > 10000 nM T17523 CND39O 44394212 IC50 = 180 nM T17523 C84JPI 44394247 IC50 > 10000 nM T17523 CA28OJ 44394273 IC50 = 32 nM T17523 CO0T1E 44394279 IC50 = 120 nM T17523 CE25XJ 44394289 EC50 = 1200 nM T17523 C0X4ZS 44394327 EC50 = 94 nM T17523 CL5BC6 44394330 IC50 > 1000 nM T17523 CU3KA2 44394460 EC50 = 36 nM T17523 C24XDE 44394498 EC50 = 36 nM T17523 CZ14XU 44394521 EC50 = 1600 nM T17523 CV9N2T 44394539 EC50 = 33000 nM T17523 C6XO8W 44394564 EC50 = 4200 nM T17523 CI75GS 44398012 EC50 = 170 nM T17523 CCFT02 44398049 EC50 = 89 nM T17523 CRYM50 44398058 EC50 = 400 nM T17523 CR3K9W 44398074 EC50 = 660 nM T17523 C4DIT3 44398076 EC50 = 160 nM T17523 C3H2IY 44398170 EC50 = 190 nM T17523 CL5SY3 44398172 EC50 = 7400 nM T17523 CR4TH0 44406004 EC50 = 1.259 nM T17523 C3JF1Q 44406009 EC50 = 63.1 nM T17523 CK6J2H 44406749 EC50 = 19.95 nM T17523 CDY46P 44412165 IC50 = 1500 nM T17523 CR2DT4 44412221 IC50 = 1000 nM T17523 CRV34X 44412232 IC50 = 300 nM T17523 CV63YC 44412233 IC50 = 1000 nM T17523 CQ1V3J 44412282 IC50 = 700 nM T17523 CB6KR7 44412294 IC50 = 540 nM T17523 CTV5M0 44412353 IC50 = 2100 nM T17523 CN7K2O 44412364 IC50 = 720 nM T17523 CL1GJ3 44412415 IC50 = 630 nM T17523 CV28IK 44412416 IC50 = 350 nM T17523 CBM50W 44412428 IC50 = 1400 nM T17523 C05TUB 44412658 EC50 > 10000 nM T17523 CH51GD 44412659 EC50 > 10000 nM T17523 C3M5SO 44412702 EC50 > 10000 nM T17523 CBUQ92 44412827 EC50 > 10000 nM T17523 CM8IK4 44412854 EC50 > 10000 nM T17523 CBL87K 44412867 EC50 > 10000 nM T17523 COA6Q1 44412868 EC50 > 10000 nM T17523 C80JSN 44412882 EC50 > 10000 nM T17523 C2WV6S 44412883 EC50 > 10000 nM T17523 C84PLZ 44412908 EC50 > 10000 nM T17523 C78DOK 44412936 EC50 > 10000 nM T17523 CH6Z8V 44412962 EC50 > 10000 nM T17523 C3MWD4 44412971 EC50 > 10000 nM T17523 CJC06H 44412994 EC50 > 10000 nM T17523 CT6EU7 44413274 IC50 = 2700 nM T17523 CYO6R3 44413349 IC50 = 32 nM T17523 CH9NL4 44413365 IC50 = 110 nM T17523 CW8E0R 44413415 IC50 = 390 nM T17523 CYW5D3 44413430 IC50 = 160 nM T17523 CJ5S2H 44413446 IC50 = 120 nM T17523 CWRZ40 44413447 IC50 = 110 nM T17523 CVC61G 44413482 IC50 = 230 nM T17523 CWL92R 44422573 EC50 = 2300 nM T17523 CW67ZB 44422578 EC50 = 440000 nM T17523 C12CHR 44422579 EC50 = 340 nM T17523 C0I3LB 44422601 EC50 = 230 nM T17523 C2O7AP 44422604 EC50 = 170 nM T17523 C07YCS 44422605 EC50 = 147 nM T17523 C7O0PC 44422606 EC50 = 150 nM T17523 C0W3FQ 44439850 IC50 > 10000 nM T17523 CB4Z3I 44439851 IC50 > 10000 nM T17523 C9SFT8 44439852 IC50 > 10000 nM T17523 CS9H0L 44517795 EC50 = 1330 nM T17523 CX13MK 44547414 EC50 = 160 nM T17523 CP18DA 44565596 IC50 = 10.3 nM T17523 CO8AD3 44565597 IC50 = 3.6 nM T17523 CS13TE 44565622 IC50 = 8.3 nM T17523 COH39N 44565714 IC50 = 5.24 nM T17523 CB1GT5 44565715 IC50 = 24.8 nM T17523 CAV3F9 44565716 IC50 = 26.9 nM T17523 C76DFZ 44565717 IC50 = 4.87 nM T17523 CMG7L1 44565738 IC50 = 11.7 nM T17523 CH8SJ9 44565739 IC50 = 1.23 nM T17523 CX9AZ4 44591249 IC50 = 4 nM T17523 C3NOY0 44591250 IC50 = 3.5 nM T17523 C3TAY6 44591264 IC50 = 1.8 nM T17523 CGCL62 44591265 IC50 = 1.1 nM T17523 C10TGI 44591266 IC50 = 1.9 nM T17523 CLTI41 44607573 IC50 = 308 nM T17523 C07PRQ 44607574 IC50 = 253 nM T17523 CF1IW9 44607575 IC50 = 163 nM T17523 C42JLY 44607576 IC50 = 417 nM T17523 C5MQ6V 44607577 IC50 = 105 nM T17523 CC9I1H 44607579 IC50 = 169 nM T17523 CX5E6T 44607580 IC50 = 89 nM T17523 CAI1Y0 44607581 IC50 = 286 nM T17523 C8X9RQ 44607582 IC50 = 302 nM T17523 C7JV5W 44620882 EC50 = 570 nM T17523 CBFP69 44620883 EC50 = 2980 nM T17523 C3CGS5 44620884 EC50 = 3900 nM T17523 CWF1P6 44620886 EC50 = 7200 nM T17523 CU9QV8 44620892 EC50 = 46 nM T17523 C71QPL 44620894 EC50 = 45 nM T17523 CP73BC 44620895 EC50 = 52 nM T17523 C6T4QB 45377662 EC50 = 106 nM T17523 C73DCB 46174905 EC50 = 420 nM T17523 CSTA18 46224712 EC50 > 10000 nM T17523 C4QB8F 46224713 EC50 > 10000 nM T17523 C4HN6L 46224714 EC50 > 10000 nM T17523 CF75RO 46224715 EC50 = 116 nM T17523 C6R9SJ 46224716 EC50 > 10000 nM T17523 CB56OX 46224767 EC50 = 100 nM T17523 CHC1D9 46224768 EC50 = 100 nM T17523 C15WRO 46224769 EC50 = 560 nM T17523 CMW59H 46225233 EC50 > 10000 nM T17523 CV5T1F 46225282 EC50 > 10000 nM T17523 CF74HE 46225283 EC50 > 10000 nM T17523 C6XAU7 46225284 EC50 > 10000 nM T17523 CL4H8B 46225285 EC50 > 10000 nM T17523 CQY5P8 46866185 EC50 = 120 nM T17523 C6LJ7A 46866186 EC50 = 140 nM T17523 CW6RX2 46881847 EC50 = 5.7 nM T17523 CAHC81 46881875 EC50 = 19 nM T17523 C0BOR7 46881876 EC50 = 800 nM T17523 CCS12Z 46881877 EC50 = 670 nM T17523 C3QMS1 46881912 EC50 = 1700 nM T17523 CTL89X 46884020 EC50 = 15.98 nM T17523 CJ21TY 46885796 IC50 = 3.4 nM T17523 CZDL71 46885798 IC50 = 6.5 nM T17523 CCX14T 49835928 EC50 = 56 nM T17523 CW9XF4 49835930 EC50 = 250 nM T17523 CS25XW 49835989 EC50 = 602 nM T17523 CX8KV1 49835990 EC50 = 1700 nM T17523 C5Z6RM 49839234 EC50 = 26 nM T17523 C4BXP1 49848557 EC50 > 39810.72 nM T17523 CMV6Y2 49868651 EC50 = 0.5 nM T17523 CH0B8K 50925337 EC50 = 0.92 nM T17523 CD2MT6 51000470 IC50 = 21 nM T17523 C9C6YQ 51057916 IC50 = 63 nM T17523 C1DYT0 53358422 IC50 = 25 nM T17523 CAOJ50 53358423 IC50 = 34 nM T17523 CC7DZ4 53362086 EC50 = 85 nM T17523 CU3Y6D 53388307 IC50 = 59 nM T17523 C03XNJ 53388308 IC50 = 75 nM T17523 CNDU92 54580601 IC50 = 6400 nM T17523 C32GIR 54580602 IC50 = 94 nM T17523 C5M2PI 54580603 IC50 = 64 nM T17523 C60WFA 54580604 IC50 = 448 nM T17523 C05AKS 54580605 IC50 = 46 nM T17523 C1VOF0 54581610 IC50 = 589 nM T17523 CJIG47 54581611 IC50 = 115 nM T17523 CTXJ83 54582605 IC50 = 52 nM T17523 CE3M4W 54582606 IC50 = 80 nM T17523 CWNO65 54582607 IC50 = 58 nM T17523 CXYR89 54582609 IC50 = 575 nM T17523 C4M8ZE 54583567 IC50 = 93 nM T17523 C1P2ZL 54584547 IC50 = 931 nM T17523 C8P2AH 54584548 IC50 = 348 nM T17523 C8GK0W 54584549 IC50 = 269 nM T17523 C47IDC 54584551 IC50 = 130 nM T17523 C7CWH4 54585466 IC50 = 34 nM T17523 CI3R5N 54585493 IC50 = 573 nM T17523 C8VHC7 54585494 IC50 = 513 nM T17523 C7E3AF 54585495 IC50 = 515 nM T17523 C7PKV6 54586461 IC50 = 8100 nM T17523 CQKD12 54586463 IC50 = 118 nM T17523 C8PKX0 54587490 IC50 = 44 nM T17523 CU62DN 54764919 EC50 > 50000 nM T17523 C1ODY4 56662043 IC50 = 211 nM T17523 CWUO23 56672438 IC50 = 2400 nM T17523 C1T9NM 56675824 IC50 = 233 nM T17523 CBP52E 56679130 IC50 = 911 nM T17523 CTI60N 56682427 IC50 = 6300 nM T17523 COPR62 56682428 IC50 = 173 nM T17523 C3Z6HO 56835136 EC50 = 54 nM T17523 C1RK0O 57390238 EC50 = 440 nM T17523 CKWG20 57390239 EC50 = 262 nM T17523 C2PNZ0 57390242 EC50 = 396 nM T17523 CT9J5U 57390243 EC50 = 68 nM T17523 CDWY69 57391736 EC50 = 3500 nM T17523 C1HQ3L 57392027 EC50 = 210 nM T17523 C2URS6 57392028 EC50 = 3100 nM T17523 CW42EG 57393480 EC50 = 2600 nM T17523 CR3ZN8 57393481 EC50 = 7300 nM T17523 C30FXU 57393538 EC50 = 208 nM T17523 C5LA3H 57393539 EC50 = 1800 nM T17523 CU4JF9 57395198 EC50 = 3100 nM T17523 C80DTW 57395199 EC50 = 2800 nM T17523 C5RLV2 57395254 EC50 = 287 nM T17523 CM74JH 57395471 EC50 = 104 nM T17523 CG0FN5 57396981 EC50 = 601 nM T17523 CU9W3T 57396983 EC50 = 1300 nM T17523 CNV5J4 57397316 EC50 = 306 nM T17523 CJS18O 57397318 EC50 = 1800 nM T17523 CDIM94 57397319 EC50 = 5400 nM T17523 CPY57D 57397320 EC50 = 72 nM T17523 C3KS0A 57397321 EC50 = 314 nM T17523 C6GH7W 57398735 EC50 = 1300 nM T17523 CCZI80 57398794 EC50 = 6000 nM T17523 CRYC82 57398795 EC50 = 2100 nM T17523 CR21DL 57398995 EC50 = 1600 nM T17523 CT7E0J 57398996 EC50 = 433 nM T17523 CXO9I1 57398998 EC50 = 147 nM T17523 C58GRL 57398999 EC50 = 660 nM T17523 CA3P8N 57400396 EC50 = 920 nM T17523 CTO8P5 57400397 EC50 = 304 nM T17523 CRNH90 57400467 EC50 = 658 nM T17523 CMNS27 57400709 EC50 = 2800 nM T17523 C49NHR 57400712 EC50 = 3200 nM T17523 CS3I9U 57400714 EC50 = 92 nM T17523 CM5L3B 57402195 EC50 = 5400 nM T17523 C3VIB7 57402197 EC50 = 4800 nM T17523 CE3CM0 57402269 EC50 = 1500 nM T17523 C9N1VH 57403951 EC50 = 220 nM T17523 C12UZA 57403952 EC50 = 2600 nM T17523 COE91B 57699087 Ki > 10000 nM T17523 C5YS7U 58329611 EC50 > 10000 nM T17523 C8FZ4S 59384310 EC50 = 4.57 nM T17523 CQ52OA 59384375 EC50 = 3.6 nM T17523 C5UTG1 66829311 EC50 > 1000 nM T17523 C6AZY0 67249162 EC50 > 10000 nM T17523 CX6SF2 67250226 EC50 = 8600 nM T17523 CY09OV 69263869 EC50 > 10000 nM T17523 CR4V0T 71450073 EC50 = 1195 nM T17523 C9IKU5 78321974 EC50 = 10.5 nM T17523 CL74JM 90309142 IC50 > 10000 nM T17523 C72NCP 118728432 IC50 > 10000 nM T17523 C9U4QR 124221654 EC50 = 154 nM T17523 C01YZA 134129958 EC50 = 694 nM T17523 C9XCH3 134129983 EC50 = 410 nM T17523 CVYH81 134130022 EC50 > 100000 nM T17523 COK2V9 134130023 EC50 = 541 nM T17523 CK3D4G 134130066 EC50 = 331 nM T17523 C9J4YQ 134130071 EC50 = 57600 nM T17523 CO7NQ6 134130111 EC50 = 1480 nM T17523 CDFI08 134130114 EC50 = 1980 nM T17523 C2XC8U 134130131 EC50 = 9250 nM T17523 CAOF06 134130145 EC50 = 470 nM T17523 CCMS20 134130146 EC50 > 100000 nM T17523 C4KI5E 134130150 EC50 = 1100 nM T17523 CUE0N7 134130169 EC50 > 100000 nM T17523 CNW53I 134130183 EC50 > 100000 nM T17523 CVA1C4 134130188 EC50 > 100000 nM T17523 CS0W9B 134130192 EC50 = 1020 nM T17523 C90GZS 134130203 EC50 > 100000 nM T17523 CYS41M 134130243 EC50 > 100000 nM T17523 C25EHG 134130292 EC50 = 1930 nM T17523 CHXD46 134130316 EC50 = 350 nM T17523 C7K1UH 134130375 EC50 = 19900 nM T17523 C4B2LQ 134130519 EC50 = 38 nM T17523 CE3O4Z 134130538 EC50 > 100000 nM T17523 C3NC1O 134130546 EC50 = 433 nM T17523 CJH4K9 134130548 EC50 > 100000 nM T17523 CD9YI4 134130571 EC50 = 816 nM T17523 C3YO7L 134130622 EC50 > 100000 nM T17523 CD7W9Y 134130662 EC50 = 115 nM T17523 C6JB4Z 134130695 EC50 = 640 nM T17523 CMX5L2 134130704 EC50 > 100000 nM T17523 CE9AV5 134130732 EC50 = 693 nM T17523 C6V4DA 134130884 EC50 = 1080 nM T17523 CGK8F7 134130947 EC50 = 2060 nM T17523 C4FBV1 134130960 EC50 > 100000 nM T17523 CFU7G1 134131038 EC50 > 100000 nM T17523 CP67CL 134131039 EC50 > 100000 nM T17523 CXKZ69 134131043 EC50 > 100000 nM T17523 CU93MF 134131067 EC50 = 1430 nM T17523 CV20CR 134131071 EC50 = 165 nM T17523 C1F7MJ 134131075 EC50 = 18300 nM T17523 C2VW9K 134131081 EC50 = 187 nM T17523 CJBU52 134131130 EC50 > 100000 nM T17523 CJI9U7 134131169 EC50 = 5070 nM T17523 CLM0H7 134131188 EC50 = 3100 nM T17523 CA86SG 134131209 EC50 = 1190 nM T17523 CX84LY 134131253 EC50 = 11100 nM T17523 C2OEB6 134131256 EC50 = 3920 nM T17523 C6GE4C 134131291 EC50 > 100000 nM T17523 CBKF68 134131297 EC50 = 724 nM T17523 CCH9O4 134131316 EC50 > 100000 nM T17523 CFR58S 134131363 EC50 = 1900 nM T17523 CNVC46 134131381 EC50 = 211 nM T17523 CE13OT 134131399 EC50 = 13500 nM T17523 CS13QG 134131470 EC50 = 3410 nM T17523 C9UB6W 134131475 EC50 = 2570 nM T17523 C64QZX 134131495 EC50 > 100000 nM T17523 C09ZOI 134131497 EC50 = 10300 nM T17523 C6DJ2N 134131598 EC50 = 1010 nM T17523 CDMT01 136042186 EC50 = 3800 nM T17523 CXF0T2 136042187 EC50 = 1000 nM T17523 CZL4I2 136042188 EC50 = 3600 nM T17523 C14VAU 136042189 EC50 = 2100 nM T17523 C0ZM4R 145966230 IC50 > 1000 nM T17523 C6JW8K 145976329 IC50 > 1000 nM T17523 CRF7V0 155317229 IC50 > 1000 nM T17523 CX76PB 155317261 IC50 > 1000 nM T17523 CW10AC 155317265 IC50 > 1000 nM T17523 C43CXP 155317276 IC50 > 1000 nM T17523 CLG86C 155317279 IC50 > 1000 nM T17523 CPY85W 16215109 EC50 = 7.4 nM T17523 CZSI05 44438257 EC50 = 347 nM T17523 CWKU57 44438259 EC50 = 16.8 nM T17523 CT3AX1 44438261 EC50 = 33.1 nM T17523 D00VHN 46905530 IC50 = 15 nM T17523 D02LTS 59393720 EC50 = 245 nM T17523 D04IAF 11452022 EC50 = 0.6 nM T17523 D04XCB 10149595 IC50 > 10000 nM T17523 D05EDD 11588811 EC50 = 500 nM T17523 D05KEE 10904818 EC50 = 1.259 nM T17523 D06DYN 9908268 EC50 = 0.09 nM T17523 D06GFH 11545181 EC50 = 6100 nM T17523 D06XMB 44394220 IC50 = 760 nM T17523 D07EAB 10215259 IC50 = 2500 nM T17523 D08VLT 10125714 IC50 > 10000 nM T17523 D0D5QS 11725751 IC50 = 26 nM T17523 D0LO4T 10287034 IC50 = 86 nM T17523 D0N0BN 44394248 IC50 = 6300 nM T17523 D0P1TY 44344193 IC50 = 140 nM T17523 D0P2AZ 10149721 IC50 = 5400 nM T17523 D0ZU0O 4077460 IC50 > 10000 nM T89658 D03VOJ 8768 IC50 = 239000 nM T89658 C54JUR 25043 IC50 = 141000 nM T89658 C70HVL 77888 IC50 = 137000 nM T89658 CPI2E4 80447 IC50 = 71600 nM T89658 C07AKH 786691 IC50 = 20000 nM T89658 CY4MC6 3505109 IC50 = 145000 nM T89658 CGN9J7 44267478 IC50 = 25000 nM T89658 CH4Q6A 145964401 IC50 = 6100 nM T89658 CHU61S 145964420 IC50 = 600 nM T89658 C6YCA8 145964710 IC50 = 700 nM T89658 CV6F7L 145966788 IC50 = 600 nM T89658 CBWX17 145967285 IC50 = 900 nM T89658 COR9X3 145972736 IC50 = 700 nM T89658 CQ0M2X 145972809 IC50 = 7500 nM T89658 CF95RZ 145972878 IC50 = 600 nM T89658 CXI0D1 145975081 IC50 = 700 nM T89658 CG84ZR 145975487 IC50 = 400 nM T89658 C91FOT 145976006 IC50 = 800 nM T89658 C3F4UH 145978039 IC50 = 500 nM T53381 D01JUF 5775 Ki = 7.6 nM T53381 D03MIR 3157 Ki = 0.3236 nM T53381 D04DKH 4418 Ki = 1.202 nM T53381 D05MBZ 129211 Ki = 0.058 nM T53381 D08JIV 2162 Ki = 5370 nM T53381 D09EBS 4636 Ki = 1348.96 nM T53381 D09MWJ 2092 Ki = 3.162 nM T53381 D0AE3X 2435 Ki = 933.25 nM T53381 D0CQ0Z 33630 Ki = 602 nM T53381 D0H4JM 8969 Ki = 1.6 nM T53381 D0O6IZ 4436 EC50 < 5011.87 nM T53381 D0P9RF 5401 Ki = 0.85 nM T53381 D0U0VU 5312125 Ki = 1.995 nM T53381 D0U3DU 5311068 Ki = 0.015 nM T53381 D0WV3U 4893 Ki = 0.17 nM T53381 D00KZF 2419 Ki = 0.778 nM T53381 D02FNU 56971 Ki = 46 nM T53381 D02LHR 33625 Ki = 110 nM T53381 D02ZSU 9838763 EC50 < 100000 nM T53381 D03QMR 5685 Ki = 0.2512 nM T53381 D04OIF 44247584 Ki = 1.1 nM T53381 D04XCQ 10099811 Ki = 340 nM T53381 D07BCO 5684 Ki = 4.571 nM T53381 D08OWQ 122295 Ki = 33 nM T53381 D0B1MJ 6918097 Ki = 79.43 nM T53381 D0L5TJ 10527469 Ki = 0.97 nM T53381 D0L9SN 4431 Ki = 0.3 nM T53381 D0N7LZ 126225 Ki = 1.6 nM T53381 D0P9FT 148842 Ki = 1.5 nM T53381 D0U3HP 164089 Ki = 0.04 nM T53381 D0Z2UD 9872515 Ki = 63.1 nM T53381 D0Z3UP 216249 EC50 > 10000 nM T53381 C5H9CN 9287 Ki > 10000 nM T53381 C28VFY 60602 Ki = 100 nM T53381 CN9GK1 104911 Ki = 5 nM T53381 CT1M8Y 119204 Ki = 630.96 nM T53381 CFD09K 121102 Ki = 0.6026 nM T53381 C2H1VA 131829 Ki = 2691.53 nM T53381 CY0O6P 151779 Ki = 309 nM T53381 CZ0D8W 180707 Ki = 331 nM T53381 CF4V5Q 185076 Ki = 562.34 nM T53381 CHLI84 210172 Ki = 1.047 nM T53381 CMV89P 671623 Ki > 940 nM T53381 C1TV2F 1070749 Ki = 30 nM T53381 CZG25W 1376848 Ki = 92 nM T53381 CLXC53 3000341 Ki = 41.7 nM T53381 CAQ2J0 3034396 Ki = 5480 nM T53381 CU4T6Q 3086326 Ki = 2398.83 nM T53381 C2ZYB3 3826471 Ki = 16.6 nM T53381 CF6IK7 3894573 Ki = 15.85 nM T53381 CC9V5K 4013695 Ki = 0.3631 nM T53381 C5K4PX 6603808 Ki = 10.47 nM T53381 CZ2M3Q 9794803 EC50 < 5011.87 nM T53381 CD47WU 9795167 EC50 = 158.49 nM T53381 CNJ92E 9797396 Ki = 69 nM T53381 CVZ64M 9798183 Ki = 22 nM T53381 CEX96I 9798656 Ki = 37 nM T53381 CN90IV 9804599 Ki = 31.62 nM T53381 C0L2CT 9808529 Ki = 38 nM T53381 CG0I2Z 9816460 EC50 = 181.97 nM T53381 C4TKB3 9816461 EC50 < 100000 nM T53381 C0HZL7 9816515 EC50 = 15.85 nM T53381 C1XA0W 9816986 EC50 < 5011.87 nM T53381 C1X0UA 9817256 Ki = 7585.78 nM T53381 CMB3R5 9824384 Ki = 0.06026 nM T53381 C6KJ7P 9827677 Ki = 150 nM T53381 CQZ6I0 9828476 Ki = 66.07 nM T53381 C0VO7E 9830292 Ki = 660 nM T53381 CH09PL 9837285 Ki = 0.45 nM T53381 CHF96B 9837963 EC50 < 100000 nM T53381 CCQ9W3 9838192 EC50 > 10000 nM T53381 C2EAU0 9838294 EC50 < 100000 nM T53381 C2O4HM 9838376 EC50 < 5011.87 nM T53381 C3XCW9 9840212 EC50 < 100000 nM T53381 CAK7C9 9844511 Ki = 177 nM T53381 C5I1XD 9847419 Ki = 115 nM T53381 CQM8A3 9847845 Ki = 0.466 nM T53381 CCB7Z6 9850782 Ki = 111 nM T53381 CY2D5T 9851486 Ki = 512.86 nM T53381 C1SEL3 9859855 EC50 = 251.19 nM T53381 CKF2T8 9864325 Ki = 0.83 nM T53381 CTY02P 9865254 Ki = 7.9 nM T53381 C40JBW 9865801 Ki = 1.259 nM T53381 C7WAK9 9872440 Ki = 73 nM T53381 CK5BJ6 9872851 Ki = 25.12 nM T53381 CS41GJ 9877827 Ki = 3.7 nM T53381 C7ER3F 9881853 EC50 < 100000 nM T53381 CV2HW7 9883506 Ki = 49.7 nM T53381 C6A9OS 9890459 Ki = 260 nM T53381 CD2KC4 9891213 Ki = 0.03981 nM T53381 CQ9WG1 9891937 Ki = 25.12 nM T53381 CM7H6I 9891967 IC50 = 13.4 nM T53381 CAM25C 9894665 Ki = 52 nM T53381 C8HS4Q 9895326 Ki = 467.74 nM T53381 C5Y2AZ 9895338 Ki = 204.17 nM T53381 CK7C9L 9903313 EC50 = 630.96 nM T53381 C8RZ7N 9903932 EC50 = 3162.28 nM T53381 CYWQ50 9906447 Ki > 10000 nM T53381 CY2I0L 9908478 Ki = 0.95 nM T53381 CI1H6U 9909211 Ki = 2.512 nM T53381 C0Y4CZ 9913449 Ki = 85 nM T53381 C5THY1 9913616 IC50 = 15.9 nM T53381 CBX74I 9915831 Ki = 75 nM T53381 CT6QX7 9916549 Ki = 290 nM T53381 CKV0N1 9920786 Ki = 1.1 nM T53381 CUI0H7 9930376 Ki = 16 nM T53381 C1C5KY 9931327 Ki = 1.9 nM T53381 C06OWM 9934955 Ki = 73 nM T53381 CUQ8I5 9947861 Ki = 2398.83 nM T53381 C4G9VQ 9954092 Ki = 0.1288 nM T53381 CD97EL 9959671 Ki = 180 nM T53381 C6LZS7 9959689 Ki = 130 nM T53381 CW89JP 9960311 Ki = 75 nM T53381 CF1C5Q 9960497 Ki = 210 nM T53381 C7JXL1 9976756 Ki = 11.48 nM T53381 C2WVQ9 9982050 Ki = 3.04 nM T53381 CF7QK6 9982585 Ki = 1100 nM T53381 C6PCS8 9984150 Ki = 1500 nM T53381 CD0IS5 9985476 Ki = 250 nM T53381 C4IG8L 10005161 Ki = 0.25 nM T53381 CA29FW 10015132 IC50 = 1122.02 nM T53381 C6XGV2 10020855 Ki = 118 nM T53381 CRH7V9 10026936 Ki = 1600 nM T53381 CGN05I 10029146 Ki = 480 nM T53381 C05ICW 10031709 Ki = 440 nM T53381 CZX09T 10038958 EC50 < 100000 nM T53381 C3A1ME 10047430 Ki = 105 nM T53381 C9P4AC 10048729 Ki = 6.59 nM T53381 C71CVU 10060965 IC50 = 416.87 nM T53381 C0I2RV 10065903 Ki = 933.25 nM T53381 CDF0Z2 10071710 Ki = 1.259 nM T53381 CN9B1F 10074286 Ki = 0.43 nM T53381 CVD98U 10083742 EC50 < 100000 nM T53381 CSW74O 10084685 EC50 < 100000 nM T53381 CC2ZY0 10089254 Ki = 794.33 nM T53381 C0IWD7 10091187 Ki = 4.49 nM T53381 C8NQ3I 10092649 Ki = 290 nM T53381 C3SJX0 10095044 Ki = 1.5 nM T53381 CP51OC 10097317 Ki = 1500 nM T53381 CLW53J 10097792 Ki = 0.2455 nM T53381 CE27RV 10135864 EC50 > 10000 nM T53381 COPD43 10160408 IC50 = 2.6 nM T53381 CSJ40T 10198532 EC50 = 10 nM T53381 CJ31LA 10199052 EC50 < 5011.87 nM T53381 C7MKP9 10199335 Ki = 2630.27 nM T53381 CU2B9P 10221004 Ki = 2238.72 nM T53381 CX9YD5 10221005 EC50 < 1995.26 nM T53381 C12UXA 10221066 EC50 < 100000 nM T53381 CO64WJ 10236758 Ki = 1000 nM T53381 CCF6U9 10244367 EC50 < 100000 nM T53381 C8SYA1 10252540 Ki = 3.236 nM T53381 C0U3WR 10314056 Ki = 1515 nM T53381 C62PAC 10318686 Ki = 65.5 nM T53381 C06YPQ 10342554 Ki = 39.5 nM T53381 CIP38T 10344976 Ki = 0.7244 nM T53381 CI17PT 10348924 Ki = 3.9 nM T53381 COC7M0 10363912 Ki = 9.333 nM T53381 C0W8QR 10364538 Ki = 3841 nM T53381 C8GR5I 10364994 Ki = 0.06761 nM T53381 CS7F3J 10371061 Ki = 340 nM T53381 CE9IN1 10378649 EC50 < 5011.87 nM T53381 C4H6YF 10379435 Ki = 3801.89 nM T53381 C3N7TF 10382537 Ki = 281.84 nM T53381 CSAF82 10393665 Ki = 80 nM T53381 CG1IR6 10394346 Ki = 20.4 nM T53381 C0MBY3 10399043 EC50 < 5011.87 nM T53381 CQ52MH 10414908 Ki = 220 nM T53381 C7Z5FO 10415038 Ki = 18 nM T53381 C9EIT6 10415156 Ki = 1280 nM T53381 CM76FU 10422033 EC50 < 5011.87 nM T53381 C0R3LA 10423384 EC50 < 100000 nM T53381 CP7B3M 10430193 Ki = 0.1514 nM T53381 CCP0S9 10434440 Ki = 0.13 nM T53381 CIQ02H 10436842 Ki = 590 nM T53381 CZTU54 10437624 Ki = 580 nM T53381 CQ93PA 10438280 Ki = 140 nM T53381 C7GEB0 10474042 Ki = 5.95 nM T53381 C0D1VZ 10479323 Ki = 19.05 nM T53381 CW16TJ 10481087 Ki = 600 nM T53381 C3MIH8 10487999 Ki = 0.78 nM T53381 C6UFO7 10506484 Ki = 1100 nM T53381 C85BUY 10506673 Ki = 65 nM T53381 CX73IB 10506729 Ki = 22 nM T53381 CY84UO 10507089 Ki = 190 nM T53381 C69OVN 10507129 Ki = 220 nM T53381 CMG18U 10507220 Ki = 700 nM T53381 C3KX6O 10507357 Ki = 407 nM T53381 C6C1NB 10507411 Ki = 1100 nM T53381 CKJI08 10507500 Ki = 330 nM T53381 CJ0K1T 10507651 Ki = 457.09 nM T53381 C2U8AC 10508016 Ki = 741.31 nM T53381 C4XZ3Y 10508132 Ki = 1698.24 nM T53381 C0U9GR 10508330 Ki = 120 nM T53381 CZP09X 10508332 Ki = 316.23 nM T53381 CR0XV8 10530491 Ki = 37 nM T53381 C35RPS 10530552 Ki = 31 nM T53381 C41XOR 10531022 Ki = 150 nM T53381 C0D4VW 10531157 Ki = 32 nM T53381 CE82ZX 10531476 Ki = 93 nM T53381 C4X9EF 10531532 Ki = 1148.15 nM T53381 CJ3CL2 10531675 Ki = 190 nM T53381 C7MI2N 10531766 Ki = 302 nM T53381 C8PA4X 10549596 Ki = 0.3715 nM T53381 CH8W9A 10554140 Ki = 21 nM T53381 CCKT30 10554745 Ki = 690 nM T53381 CPE27N 10554913 Ki = 37 nM T53381 C8NXE5 10554957 Ki = 680 nM T53381 C2ONS3 10555024 Ki = 620 nM T53381 CV7F9T 10555223 Ki = 2600 nM T53381 C16APC 10555288 Ki = 180 nM T53381 C7ROD9 10556164 Ki = 390 nM T53381 C7LWD8 10578548 Ki = 1100 nM T53381 C93CLB 10578715 Ki = 16 nM T53381 C18HKX 10578735 Ki = 480 nM T53381 CT0ML5 10578926 Ki = 1700 nM T53381 C4SVP1 10578990 Ki = 72 nM T53381 CF24MW 10579368 Ki = 1737.8 nM T53381 C2LRK3 10579632 Ki = 120 nM T53381 CFQB52 10580182 Ki = 5370 nM T53381 CZ8IX1 10602912 Ki = 137 nM T53381 CR8ZX2 10603727 Ki = 398 nM T53381 CD7W1O 10603739 Ki = 87 nM T53381 CK8SO7 10603951 Ki = 501.19 nM T53381 C2G4IR 10617200 Ki = 7.943 nM T53381 C8B5CJ 10621590 Ki = 16.6 nM T53381 CE5CU8 10621592 Ki = 79.43 nM T53381 CC34GW 10626453 Ki = 1600 nM T53381 CY4H5J 10626493 Ki = 250 nM T53381 COU08R 10626610 Ki = 370 nM T53381 C6BHD5 10626686 Ki = 63 nM T53381 CNE1X0 10626726 Ki = 14 nM T53381 CUF48J 10626772 Ki = 480 nM T53381 CVG42P 10626843 Ki = 79 nM T53381 CQ13HM 10626910 Ki = 124 nM T53381 CXD31C 10626911 Ki = 51 nM T53381 CB26QH 10626982 Ki = 436.52 nM T53381 CYG6R7 10627003 Ki = 41 nM T53381 CSWC40 10627021 Ki = 316.23 nM T53381 CFA2R6 10627090 Ki = 260 nM T53381 C3TSO7 10627094 Ki = 910 nM T53381 CDC19N 10627155 Ki = 30 nM T53381 CF38IK 10627279 Ki = 270 nM T53381 CZ3T7S 10627329 Ki = 120 nM T53381 CER8L0 10640982 Ki = 199.53 nM T53381 C70QNW 10649481 Ki = 200 nM T53381 C9VY7F 10650129 Ki = 65 nM T53381 C6J4OK 10650633 Ki = 180 nM T53381 C4HP6A 10650726 Ki = 14 nM T53381 CLV1Q4 10650843 Ki = 55 nM T53381 CF1P6Z 10651080 Ki = 1148.15 nM T53381 CBN78H 10651219 Ki = 140 nM T53381 CV2HA5 10651636 Ki = 250 nM T53381 C3K7UP 10651654 Ki = 323.59 nM T53381 CU7W3E 10655390 Ki = 0.17 nM T53381 C7ZUW0 10657835 Ki = 0.35 nM T53381 C07UGY 10673657 Ki = 340 nM T53381 CG6P7N 10674055 Ki = 10 nM T53381 C35NWA 10674133 Ki = 137 nM T53381 CRQD91 10674333 Ki = 290 nM T53381 CX69JL 10674544 Ki = 1560 nM T53381 CQ9JN3 10674564 Ki = 15 nM T53381 C4EC8H 10674791 Ki = 170 nM T53381 C95VPX 10674840 Ki = 40 nM T53381 CTB7L2 10674896 Ki = 380.19 nM T53381 CC8IT7 10675068 Ki = 180 nM T53381 C92LVP 10678591 Ki = 8.7 nM T53381 C92HXV 10678895 Ki = 3.6 nM T53381 CBEP65 10688604 Ki = 16.22 nM T53381 CB0F2I 10697623 Ki = 630 nM T53381 CA80KS 10697912 Ki > 4000 nM T53381 C16NJO 10698141 Ki = 52 nM T53381 C6PVI9 10698570 Ki = 28 nM T53381 C4XZM6 10698974 Ki = 2260 nM T53381 CI4V5M 10699164 Ki = 12 nM T53381 C36PSB 10706270 Ki = 0.18 nM T53381 C0HO7D 10720893 Ki = 150 nM T53381 C87QBC 10721171 Ki = 120 nM T53381 C5WR2P 10721476 Ki = 210 nM T53381 C3WQ9B 10721564 Ki = 170 nM T53381 CZI63U 10721568 Ki = 28 nM T53381 C5L4AS 10721730 Ki = 1940 nM T53381 CPF96G 10722045 Ki = 180 nM T53381 C6N7CQ 10722099 Ki = 140 nM T53381 CE2GK7 10739024 Ki = 250 nM T53381 C1QZ3O 10743042 Ki = 11.9 nM T53381 CGQ8I3 10744391 Ki = 410 nM T53381 CU6HM4 10745305 Ki = 610 nM T53381 CHT1L0 10745380 Ki = 31 nM T53381 C1RZU6 10745566 Ki = 1900 nM T53381 CA17HU 10745664 Ki = 340 nM T53381 CW91BJ 10745766 Ki = 140 nM T53381 C6IG0M 10745901 Ki = 34 nM T53381 CS3ON2 10746137 Ki = 930 nM T53381 CJ8VM0 10747021 Ki = 560 nM T53381 CBZP19 10747201 Ki = 190 nM T53381 C51YSW 10764133 Ki = 263.03 nM T53381 CFM65K 10767981 Ki = 1.585 nM T53381 C0WMG4 10768610 Ki = 540 nM T53381 C58CRB 10768829 Ki = 9.8 nM T53381 CV1JT2 10769037 Ki = 230 nM T53381 C63FIL 10769058 Ki = 230 nM T53381 CT1K3B 10769331 Ki = 125.89 nM T53381 C6JG4Z 10769621 Ki = 780 nM T53381 CV6T3C 10770007 Ki = 91 nM T53381 C8LZM3 10770057 Ki = 51 nM T53381 C9ARF0 10770317 Ki = 152 nM T53381 C0ZPA5 10782052 Ki = 0.07 nM T53381 CS8QR2 10787126 Ki = 7.413 nM T53381 CMU59N 10791843 Ki = 710 nM T53381 C4XK8Y 10792591 Ki = 230 nM T53381 CS24OF 10792897 Ki = 54 nM T53381 C6F5HP 10792898 Ki = 62 nM T53381 CN71ZB 10793023 Ki = 320 nM T53381 C3O7YN 10793665 Ki = 446.68 nM T53381 CTXB06 10793720 Ki = 56 nM T53381 C0D6MW 10793963 Ki = 144.54 nM T53381 C6EWQ3 10811627 Ki = 1435 nM T53381 CXU6D7 10815549 Ki = 220 nM T53381 CN6ZP7 10815593 Ki = 240 nM T53381 C4ZNR1 10816815 Ki = 910 nM T53381 C68UVF 10816832 Ki = 1700 nM T53381 CO73GU 10816903 Ki = 610 nM T53381 CID39T 10817365 Ki = 110 nM T53381 CBO8N9 10818003 Ki = 346.74 nM T53381 CFC95U 10834793 Ki = 0.4898 nM T53381 C5NFU1 10836245 Ki = 18 nM T53381 CIY58E 10839105 Ki = 590 nM T53381 CKS74R 10839106 Ki = 600 nM T53381 C5SC1X 10839825 Ki = 2200 nM T53381 CP78AK 10840177 Ki = 480 nM T53381 C49YSD 10840781 Ki = 1800 nM T53381 C4LV0H 10841070 Ki = 110 nM T53381 CE80NV 10841190 Ki = 489.78 nM T53381 C2RXD0 10841296 Ki = 570 nM T53381 CYSL64 10841387 Ki = 616 nM T53381 C8TED5 10841819 Ki = 5280 nM T53381 CO9WP2 10841851 Ki = 1100 nM T53381 C70LSM 10880840 Ki = 549.54 nM T53381 C3I1CT 10892762 Ki = 142 nM T53381 CEUD36 10893672 Ki = 17.69 nM T53381 C8VT6G 10916464 Ki = 870.96 nM T53381 CBH30I 10916771 Ki = 11.78 nM T53381 CD7QW2 10917316 Ki = 5.34 nM T53381 CH95TI 10923927 Ki < 15848.93 nM T53381 C4GCP7 10928161 Ki = 35.48 nM T53381 C0N6KJ 10928520 Ki = 1.07 nM T53381 C3CI6Z 10934575 EC50 = 0.912 nM T53381 C8LPD2 10939209 Ki = 60.26 nM T53381 CTO4Z9 10949698 Ki = 34.45 nM T53381 C58LAV 10950355 Ki = 245.47 nM T53381 CAIJ61 10961351 Ki = 0.49 nM T53381 CW6T1N 10971791 Ki = 0.4074 nM T53381 CX5M6J 10974101 Ki = 4.2 nM T53381 CC2NG9 10994812 Ki = 3.92 nM T53381 C2BF0W 11014848 Ki = 3.2 nM T53381 CGW87Y 11034737 EC50 = 43.65 nM T53381 CZM27Y 11039289 Ki = 3.5 nM T53381 CH9O0P 11046644 Ki = 12.57 nM T53381 C48QYR 11058166 Ki = 912.01 nM T53381 C7JI1M 11059195 Ki < 15848.93 nM T53381 C7R2AZ 11079593 Ki = 1621.81 nM T53381 CUZ38C 11081136 Ki = 2.92 nM T53381 C91BKL 11090351 Ki = 3467.37 nM T53381 CF32NC 11092254 Ki = 0.41 nM T53381 CFE1M7 11097789 Ki = 5.012 nM T53381 CTG4I5 11098175 EC50 = 5.012 nM T53381 C84VUJ 11108001 EC50 = 7.943 nM T53381 CR6K4V 11109088 EC50 = 2.692 nM T53381 CJT65Y 11123606 Ki = 4.32 nM T53381 CF68CS 11133288 Ki = 3.631 nM T53381 C7MD3R 11133868 Ki = 22.91 nM T53381 C3ZJK1 11134424 Ki = 0.25 nM T53381 CC0HY8 11135150 Ki = 181.97 nM T53381 CG40BP 11140345 EC50 = 33.88 nM T53381 CO0XW1 11140347 Ki = 6.166 nM T53381 CA7Y5Z 11144555 Ki = 11.79 nM T53381 C73DFT 11145007 Ki = 5.96 nM T53381 CUNH28 11152823 Ki = 199.53 nM T53381 C7VKQ5 11164948 Ki = 1148.15 nM T53381 C4J8YG 11211017 Ki = 14 nM T53381 CLYZ97 11234093 Ki = 16.22 nM T53381 C90UKI 11281005 Ki = 338.84 nM T53381 CR2DJ1 11282574 Ki = 24.55 nM T53381 CH9X5G 11304777 Ki > 124 nM T53381 CCQ0S5 11338016 Ki = 15.85 nM T53381 CT3V5I 11338314 Ki = 5.6 nM T53381 C7KX6F 11430126 Ki = 0.4898 nM T53381 C7EVT0 11430491 Ki = 0.389 nM T53381 CM8I7N 11454386 Ki = 0.8913 nM T53381 C8TDA7 11488170 Ki = 199.53 nM T53381 CTMH12 11505007 Ki = 0.35 nM T53381 CS20NG 11519153 Ki = 2 nM T53381 CI8GN0 11532563 Ki = 0.3162 nM T53381 C0MF3O 11539392 Ki = 0.1259 nM T53381 COC6U3 11554541 Ki = 0.05012 nM T53381 C2IE4D 11583392 Ki = 0.03162 nM T53381 CJW9E6 11604548 Ki = 0.0631 nM T53381 C6JRN0 11619713 Ki = 0.912 nM T53381 C3IHP8 11626704 Ki = 0.05012 nM T53381 C9VAI5 11633517 Ki = 0.1995 nM T53381 CL6XP8 11638677 Ki = 1.259 nM T53381 CZA0M9 11653915 Ki = 17.5 nM T53381 C9I7KB 11669646 Ki = 0.1 nM T53381 CUVL17 11705133 Ki = 1.995 nM T53381 C7RAS6 11712250 Ki = 0.2512 nM T53381 C7PK3H 11712470 Ki = 0.0631 nM T53381 CR1L6N 11732516 Ki > 10 nM T53381 C12YTV 11742585 Ki = 3250 nM T53381 CJ60OP 11742834 Ki = 0.08913 nM T53381 C3G4FS 11751173 Ki = 0.9333 nM T53381 CO50RT 11757736 Ki = 640 nM T53381 C90XQT 11762075 Ki = 19.95 nM T53381 C06HZD 11782656 Ki = 83.24 nM T53381 C28UNM 11784634 Ki = 389.05 nM T53381 C4VL6W 11801214 Ki = 52 nM T53381 CFTI34 11801828 Ki = 1513.56 nM T53381 C4ZXG0 11801861 Ki = 14700 nM T53381 C2RPQ0 11802456 Ki = 91 nM T53381 C1VWL5 11811395 Ki = 2818.38 nM T53381 CUB53N 11857638 Ki = 0.77 nM T53381 C29HBR 11857639 Ki = 7.3 nM T53381 C29FMG 11857709 Ki = 2.2 nM T53381 CX50UR 11857710 Ki = 2.6 nM T53381 CW6V5E 11857711 Ki = 2.1 nM T53381 CD50HW 11857791 Ki = 3 nM T53381 CGL5D9 11857792 Ki = 1.6 nM T53381 CE0U9G 11857793 Ki = 0.98 nM T53381 CYJ5I7 11857794 Ki = 5.9 nM T53381 C9S5NU 11857861 Ki = 5.5 nM T53381 CU83FA 11857862 Ki = 4.1 nM T53381 CUO32E 11857863 Ki = 12 nM T53381 CD7O6J 11857864 Ki = 1.6 nM T53381 CH1WZ3 11984570 Ki = 0.09 nM T53381 CJP2T4 11994550 Ki = 15.85 nM T53381 CHE4O6 11994665 Ki = 3.388 nM T53381 C0ZRF5 11994667 Ki = 15.14 nM T53381 CQW63S 11994668 Ki = 53.7 nM T53381 CVNL73 11994670 Ki = 363.08 nM T53381 C1BZQ0 11994673 Ki = 147.91 nM T53381 CB3DJ5 11994797 Ki = 14.45 nM T53381 C1KQO2 11994915 Ki = 213.8 nM T53381 CU17YO 11995033 Ki = 28.84 nM T53381 C3F1BT 11995035 Ki = 954.99 nM T53381 C8W5JG 12039032 Ki = 6043 nM T53381 CY8DS2 12134985 Ki > 10000 nM T53381 C4CI5P 12134986 Ki = 272 nM T53381 CS6BU1 12134987 Ki = 1517 nM T53381 CPX75G 12134991 Ki > 5000 nM T53381 CI52SU 12134994 Ki = 262 nM T53381 C8WEX1 12134995 Ki = 138 nM T53381 C6S9BY 12134996 Ki = 23 nM T53381 C2U3RT 12764879 EC50 = 7360 nM T53381 C0B1QO 12764880 EC50 > 10000 nM T53381 CMA46J 13305910 Ki = 0.5129 nM T53381 C4XD7S 13442845 Ki = 160 nM T53381 C0TP9W 13442851 Ki > 940 nM T53381 CN2ZQ5 13911290 Ki = 0.308 nM T53381 CV08GM 14378574 Ki = 25 nM T53381 C4E7NH 14423371 Ki = 0.195 nM T53381 CMO81H 14925759 Ki = 91.2 nM T53381 CQ5ZJ2 15546405 Ki = 650 nM T53381 C1CX2S 15675860 Ki = 5011.87 nM T53381 CRTO23 15840661 Ki = 31.62 nM T53381 CT03WI 16040907 Ki = 8.7 nM T53381 CW5NS1 16041090 Ki = 20 nM T53381 C03VCW 16041091 Ki = 15 nM T53381 CM3O4Z 16041092 Ki = 1.6 nM T53381 CUL5M9 16041263 Ki = 3 nM T53381 C6S8AM 16041264 Ki = 1.5 nM T53381 CYTD80 16041265 Ki = 2.6 nM T53381 C86MYV 16041449 Ki = 3.7 nM T53381 CHF7K6 16041451 Ki = 2.7 nM T53381 CCJ65Y 16041628 Ki = 2.7 nM T53381 CE2Z7Y 16041629 Ki = 1.2 nM T53381 CRJX49 16041630 Ki = 4.8 nM T53381 CDTN28 16121006 Ki = 6.607 nM T53381 C1YWG6 16215415 Ki = 275 nM T53381 CNF70V 16220269 IC50 = 13800 nM T53381 CZ2IS9 16660294 Ki > 10000 nM T53381 CZ8S6B 16721032 Ki = 4.786 nM T53381 C7KS8E 16721110 Ki = 0.166 nM T53381 CHRG71 16738927 IC50 = 25.12 nM T53381 C3GD2P 17753379 Ki = 0.75 nM T53381 CM60NI 17804479 EC50 = 364 nM T53381 CN0CH5 18187410 Ki = 16 nM T53381 CT3OK4 18738380 Ki = 253 nM T53381 CF1DM9 18738384 Ki = 47 nM T53381 CEP14V 18738385 Ki = 92 nM T53381 CM6YI0 18738386 Ki = 25 nM T53381 CCO79B 18738387 Ki = 12 nM T53381 C9E4ID 18738412 Ki = 3064 nM T53381 CYT58A 19085820 Ki = 351 nM T53381 CHM64Z 19085827 Ki = 2750 nM T53381 CV8X0D 19085829 Ki = 71 nM T53381 C9CL0I 19085832 Ki = 224 nM T53381 C2EYW8 19085836 Ki = 1019 nM T53381 C6KSV0 19085839 Ki = 644 nM T53381 CRU75T 19085858 Ki = 59 nM T53381 CN5XJ1 19085866 Ki = 41 nM T53381 C2L1IX 19085869 Ki = 136 nM T53381 C4V1LT 19085876 Ki = 25 nM T53381 C7A2EC 19085881 Ki = 75 nM T53381 C8RDC1 19085894 Ki = 210 nM T53381 CC1Y7N 19085914 Ki = 76 nM T53381 C7T6HA 19085921 Ki = 3429 nM T53381 C7M9NZ 19085926 Ki = 73 nM T53381 C4F1GZ 19961018 Ki = 0.96 nM T53381 CQC2R0 19961030 Ki = 2.1 nM T53381 C4GM9S 20750645 Ki = 339 nM T53381 C3T5HF 21509921 Ki = 588.84 nM T53381 CD9Y0E 21712258 Ki = 1400 nM T53381 CT7XG9 21830793 Ki > 10000 nM T53381 C21LHM 22493224 EC50 = 79.43 nM T53381 C4UYD5 22493225 EC50 < 5011.87 nM T53381 C9V4MO 22493231 EC50 = 398.11 nM T53381 CKB2N6 22493233 EC50 < 100000 nM T53381 C0P2UY 22493236 EC50 = 3.981 nM T53381 C02AEX 22493245 Ki = 1380.38 nM T53381 CWT85U 22493254 EC50 < 5011.87 nM T53381 CK8GD3 22493257 EC50 < 5011.87 nM T53381 C09UWJ 22493258 EC50 = 19.95 nM T53381 C6BTO5 22493263 EC50 = 125.89 nM T53381 C7NGV2 22493265 EC50 = 251.19 nM T53381 CJ1G5C 22493269 EC50 < 100000 nM T53381 CR63XU 22493272 EC50 < 5011.87 nM T53381 CGI40S 22493274 EC50 < 5011.87 nM T53381 C3JW1Q 22493280 EC50 = 2.884 nM T53381 CG28DA 22493287 EC50 < 100000 nM T53381 CYHG72 22493289 EC50 = 81.28 nM T53381 CMS13N 22493316 EC50 < 100000 nM T53381 C6ADV8 22493318 EC50 = 16.22 nM T53381 CS4EI0 22493320 EC50 = 199.53 nM T53381 CSF43L 22493325 EC50 < 5011.87 nM T53381 C1QOL5 22493343 EC50 = 63.1 nM T53381 CKIJ24 22493344 EC50 < 100000 nM T53381 C7FCZ5 22493347 EC50 < 5011.87 nM T53381 CDE4R9 22493349 EC50 < 100000 nM T53381 CSCP16 22493352 EC50 = 5.012 nM T53381 C3N9RK 22493356 EC50 < 100000 nM T53381 C7XEF1 22493359 EC50 < 5011.87 nM T53381 C5ZNB0 22493365 EC50 = 19.95 nM T53381 CI1GH6 22493367 EC50 = 398.11 nM T53381 C86PSG 22493372 EC50 < 5011.87 nM T53381 CI42EA 22493379 EC50 = 316.23 nM T53381 CY80ON 22493381 EC50 < 100000 nM T53381 C4LJO9 22493387 EC50 < 100000 nM T53381 CP34UB 22493392 EC50 = 41.69 nM T53381 C9DS1F 22493401 EC50 < 5011.87 nM T53381 CAFG09 22493408 EC50 < 5011.87 nM T53381 C9T5VN 22493411 EC50 < 5011.87 nM T53381 CM86HE 22493415 EC50 = 28.84 nM T53381 CDC91N 24839550 Ki < 10000 nM T53381 CX6R0P 24894141 Ki = 56.23 nM T53381 C5QG6V 24894147 Ki = 0.4898 nM T53381 CW2FG9 24897950 Ki = 0.955 nM T53381 C13JLE 24900426 IC50 = 158.49 nM T53381 C1U9VL 24900685 IC50 = 199.53 nM T53381 CU3F7K 24900689 EC50 = 125.89 nM T53381 CPLO51 24900749 IC50 = 251.19 nM T53381 CX69CF 24900750 IC50 = 158.49 nM T53381 CE5W9U 24900751 IC50 = 31.62 nM T53381 CQDR84 24900811 IC50 = 100 nM T53381 CIL8Q7 24900812 IC50 = 316.23 nM T53381 C9YUP8 24900813 IC50 = 79.43 nM T53381 C63ILV 24900872 IC50 = 251.19 nM T53381 CSF3J2 24900874 IC50 = 630.96 nM T53381 C4AT0P 24900937 IC50 = 1000 nM T53381 C2NR7M 24900942 IC50 = 25.12 nM T53381 CW0QV2 24901141 IC50 = 63.1 nM T53381 CHWE43 24901143 IC50 = 158.49 nM T53381 C5ZCX4 24901144 IC50 = 125.89 nM T53381 CNP40V 24901209 IC50 = 398.11 nM T53381 C7MGC9 24901210 IC50 = 50.12 nM T53381 CS6BH7 24901211 IC50 = 79.43 nM T53381 C4JB7G 24901283 IC50 = 501.19 nM T53381 CBS0V5 24901284 IC50 = 39.81 nM T53381 C83MAF 24901285 IC50 = 39.81 nM T53381 CVE24O 24901347 IC50 = 12.59 nM T53381 CV5GY0 24901348 IC50 = 79.43 nM T53381 CFZ5D7 24901349 IC50 = 50.12 nM T53381 CCMQ16 24901351 IC50 = 7.943 nM T53381 CGW2U6 24901413 IC50 = 100 nM T53381 COY5H0 24901416 IC50 = 199.53 nM T53381 C1VRJ3 25014630 IC50 = 2200 nM T53381 CNLQ36 25025048 Ki = 2.6 nM T53381 C4QIC2 25025052 Ki = 10 nM T53381 C07RQX 25025053 Ki = 52 nM T53381 CB8L2N 25025244 Ki = 0.86 nM T53381 CJOY17 25066019 EC50 > 10000 nM T53381 CF7P2A 25130875 Ki = 97.72 nM T53381 C7P1QS 25130876 Ki = 16.22 nM T53381 C6G5BO 25130877 Ki > 1000 nM T53381 CL8GD3 25130878 Ki = 72.44 nM T53381 CT78MG 25130879 Ki = 43.65 nM T53381 C7WXA2 25131192 Ki > 1000 nM T53381 C3UVA0 25131193 Ki = 66.07 nM T53381 C0GM3L 25131196 Ki > 1000 nM T53381 CFUT35 25131198 Ki = 3.631 nM T53381 C1Y3TS 25131871 Ki > 1000 nM T53381 CFJ6Y9 25131876 Ki = 1.148 nM T53381 CNQX42 25132217 Ki = 354.81 nM T53381 C7WE4Y 25132564 Ki > 1000 nM T53381 C6K1TB 25132565 Ki = 154.88 nM T53381 CJ19KC 25132566 Ki = 31.62 nM T53381 CNO83H 25181488 Ki = 1.148 nM T53381 CEYF08 25181489 Ki = 3.236 nM T53381 CJ3NP5 42636941 IC50 = 204.17 nM T53381 CW2DP3 44123711 Ki > 1000 nM T53381 C2HPM1 44213730 Ki = 63.1 nM T53381 C2DS9L 44213782 Ki = 1800 nM T53381 CTR42S 44219718 EC50 > 2600 nM T53381 CB2HY8 44219719 EC50 > 10000 nM T53381 C4T7ZI 44222842 Ki = 26.3 nM T53381 C9ROX7 44267817 Ki = 4500 nM T53381 C0L4TU 44267884 Ki = 108 nM T53381 CF2DH7 44267890 Ki = 5350 nM T53381 CEL7U6 44267912 Ki = 10000 nM T53381 CF51JW 44268966 Ki = 7.15 nM T53381 C89FEL 44269124 IC50 = 323.59 nM T53381 CVE83T 44271661 EC50 = 0.5012 nM T53381 C7P2AH 44271931 EC50 < 100000 nM T53381 CSQ5L6 44271932 EC50 = 199.53 nM T53381 C5UA4W 44273916 Ki = 9 nM T53381 CMH52E 44275255 Ki = 446.68 nM T53381 C7Q2JD 44275526 Ki = 891.25 nM T53381 CPK7B3 44284333 Ki < 1000 nM T53381 CZPD80 44288485 Ki = 960 nM T53381 C5UIM4 44288492 Ki = 1500 nM T53381 CL3RI0 44288729 Ki > 5000 nM T53381 CTR4Z6 44288740 Ki = 3300 nM T53381 C4K6RC 44288741 Ki = 3400 nM T53381 CQP9B7 44288754 Ki = 1700 nM T53381 CZ5P6U 44288769 Ki = 1155 nM T53381 CV8G1J 44288792 Ki = 1300 nM T53381 CQ40MA 44288794 Ki = 2300 nM T53381 CX7BT8 44288810 Ki = 3300 nM T53381 CA16JS 44288815 Ki = 1100 nM T53381 C4KND2 44288816 Ki = 2500 nM T53381 CT7IB6 44288841 Ki = 230 nM T53381 CEM2T4 44288843 Ki > 5000 nM T53381 CZ7O4D 44288847 Ki > 5000 nM T53381 C8EJ9B 44288857 Ki = 6300 nM T53381 CKA01M 44288858 Ki > 5000 nM T53381 CL4X9R 44288864 Ki > 5000 nM T53381 C6DYQ1 44288874 Ki = 588 nM T53381 CAG7E1 44288877 Ki > 5000 nM T53381 CQ74LV 44288917 Ki = 1050 nM T53381 CQ3Y5R 44288945 Ki = 200 nM T53381 CZDR39 44288995 Ki = 2400 nM T53381 C92FEY 44289026 Ki = 3200 nM T53381 C9HMK3 44289034 Ki = 2700 nM T53381 C5ZL4A 44289035 Ki = 880 nM T53381 C71XMR 44289047 Ki = 3600 nM T53381 CW5C4G 44289058 Ki = 2900 nM T53381 C62NWB 44289089 Ki = 1300 nM T53381 C37GEA 44289100 Ki = 250 nM T53381 C1ES5Y 44289103 Ki = 682 nM T53381 CZS9B7 44289107 Ki = 330 nM T53381 CZSM05 44289112 Ki = 710 nM T53381 C51NLQ 44289248 Ki = 0.4365 nM T53381 CWC49F 44289261 Ki = 16.98 nM T53381 C14WMG 44289321 Ki = 36 nM T53381 CQW1Z3 44289344 Ki = 128 nM T53381 CFO29U 44289346 Ki > 5000 nM T53381 C1JX5M 44289437 Ki = 0.182 nM T53381 CF1UW9 44294569 Ki = 0.93 nM T53381 CBS42M 44294957 Ki = 180 nM T53381 CW6D7V 44294958 Ki = 690 nM T53381 CMQ6G5 44295044 Ki = 1100 nM T53381 C9XAB7 44295046 Ki = 420 nM T53381 C9MQ4B 44295133 Ki = 130 nM T53381 CNQ82T 44295170 Ki = 1300 nM T53381 C9Y3GE 44295192 Ki = 340 nM T53381 C4KB8E 44295193 Ki = 1900 nM T53381 C9UW2H 44295218 Ki = 420 nM T53381 CWJ13T 44298447 Ki = 2.512 nM T53381 C0F8LH 44298611 Ki = 5.012 nM T53381 C17AXP 44298626 Ki = 7.943 nM T53381 CA19EZ 44298644 Ki = 125.89 nM T53381 C0QLW1 44298650 Ki = 25.12 nM T53381 CO6K1V 44298664 Ki = 1.995 nM T53381 CMI12L 44298671 Ki = 31.62 nM T53381 CBJ31S 44298694 Ki = 19.95 nM T53381 CUO47C 44298734 Ki = 50.12 nM T53381 C4N1EM 44298746 Ki = 15.85 nM T53381 C1H2MT 44298762 Ki = 100 nM T53381 C3X6RY 44298770 Ki = 10 nM T53381 C9TR2K 44298780 Ki = 125.89 nM T53381 CX90HD 44299835 Ki = 550 nM T53381 C6HO4W 44299945 Ki = 95 nM T53381 CG82KA 44299973 Ki = 5.4 nM T53381 CL62DY 44299974 Ki = 39 nM T53381 C0LF1S 44299975 Ki = 7.5 nM T53381 CY8J6F 44300087 Ki = 31 nM T53381 CYV46S 44300107 Ki = 97 nM T53381 CLHT17 44300111 Ki = 320 nM T53381 C2WP7S 44300129 Ki = 500 nM T53381 CH59JV 44300159 Ki = 660 nM T53381 C8K3AP 44300165 Ki = 16 nM T53381 CSA23P 44300166 Ki = 170 nM T53381 C3YDV9 44300170 Ki = 11 nM T53381 CW56GZ 44301572 Ki > 5000 nM T53381 CH34AY 44301573 Ki = 4100 nM T53381 CIPQ70 44301680 Ki > 5000 nM T53381 C5EZ6B 44301681 Ki = 4800 nM T53381 CND82T 44307780 Ki = 315.8 nM T53381 C6R2DV 44308443 Ki = 13 nM T53381 C8M4HW 44308466 Ki = 15 nM T53381 CPUO39 44308654 Ki = 130 nM T53381 C6G8ZC 44311789 Ki = 41686.94 nM T53381 C5L1WN 44312036 Ki = 5011.87 nM T53381 CT46CK 44312037 Ki = 27542.29 nM T53381 C3XFH4 44312198 Ki = 102329.3 nM T53381 CKU7Y6 44316072 Ki = 44 nM T53381 CG2UB8 44316098 Ki = 52 nM T53381 C2PR8V 44318000 Ki = 4142 nM T53381 CZ5M4K 44318075 Ki = 285 nM T53381 C8JKO2 44318081 Ki = 320 nM T53381 C3J9XH 44324405 Ki = 69 nM T53381 CGP40I 44329083 EC50 < 5011.87 nM T53381 CES26R 44329133 EC50 = 15.85 nM T53381 CR3N5S 44329318 EC50 < 5011.87 nM T53381 CZ21VE 44329481 EC50 < 5011.87 nM T53381 C4ZV9T 44329701 EC50 = 251.19 nM T53381 CBZ84S 44329703 EC50 < 5011.87 nM T53381 CQY03V 44329738 EC50 < 5011.87 nM T53381 C7Z2HM 44329739 EC50 < 5011.87 nM T53381 CS2WN0 44329788 EC50 < 5011.87 nM T53381 C5AG1U 44329790 EC50 = 63.1 nM T53381 C14RBX 44329796 EC50 = 15.85 nM T53381 CG60QK 44329797 IC50 = 1995.26 nM T53381 C6US9E 44330880 Ki = 60 nM T53381 C2N0GV 44331079 Ki = 200 nM T53381 C02JUQ 44331090 Ki = 136 nM T53381 CU2H1F 44331136 Ki = 53 nM T53381 C5SLE2 44331150 Ki = 24 nM T53381 CK5R0A 44331169 Ki = 94 nM T53381 CGJB37 44331174 Ki = 149 nM T53381 CI9UV3 44331198 Ki = 99 nM T53381 C4RJ7I 44331277 Ki = 67 nM T53381 CO5T9G 44343173 EC50 < 5011.87 nM T53381 C0DS6V 44343235 EC50 < 100000 nM T53381 CK1QJ5 44343236 EC50 = 100 nM T53381 CV5N1T 44343243 EC50 < 5011.87 nM T53381 C84GDJ 44343244 EC50 = 31.62 nM T53381 CV8LE9 44343245 EC50 < 5011.87 nM T53381 CX8J0Y 44343247 EC50 = 79.43 nM T53381 C71WZX 44343251 EC50 < 100000 nM T53381 C19JFN 44343257 IC50 = 933.25 nM T53381 C17HRU 44343275 EC50 < 251.19 nM T53381 C6ZU5G 44343410 EC50 = 19.95 nM T53381 CQR12J 44343520 EC50 < 5011.87 nM T53381 CFQ32B 44343524 EC50 < 100000 nM T53381 CZ2X3A 44352155 EC50 = 794.33 nM T53381 C3I9DE 44358574 Ki = 12.65 nM T53381 C2WYI7 44361064 Ki = 436.52 nM T53381 C8OM7A 44362013 EC50 < 100000 nM T53381 CK6S1Y 44362145 EC50 < 100000 nM T53381 C7FHB4 44362146 EC50 = 12.59 nM T53381 CSFJ14 44362149 EC50 = 25.12 nM T53381 CEZ8K0 44362150 EC50 < 100000 nM T53381 CK8U9S 44362185 EC50 = 158.49 nM T53381 CHL40X 44362194 EC50 = 5.012 nM T53381 C3CF8S 44362195 EC50 = 6.31 nM T53381 C78CEY 44362196 EC50 = 31.62 nM T53381 C3AU6V 44362208 EC50 = 15.85 nM T53381 CH9B3A 44362286 EC50 < 100000 nM T53381 CF6H7S 44362287 EC50 < 100000 nM T53381 CI6DH4 44362288 EC50 < 100000 nM T53381 C2SBP1 44362289 EC50 < 100000 nM T53381 CH79ZL 44362510 EC50 < 100000 nM T53381 C0GR4S 44362511 EC50 < 100000 nM T53381 C1U0TR 44362523 EC50 < 100000 nM T53381 CEQD62 44362541 EC50 < 100000 nM T53381 CU0E7G 44362633 Ki = 2100 nM T53381 C94ORM 44362867 Ki = 750 nM T53381 CZ1KQ9 44369351 EC50 = 18.2 nM T53381 C1Y7OL 44369431 EC50 = 48.98 nM T53381 C03STZ 44369434 EC50 < 1995.26 nM T53381 C6W2MT 44369646 EC50 < 100000 nM T53381 CDR8C3 44369647 EC50 < 100000 nM T53381 C27FZA 44417706 Ki = 416.87 nM T53381 C31WOV 44417713 Ki = 22.39 nM T53381 C85GUJ 44420408 Ki = 1.549 nM T53381 CHIA46 44420412 Ki = 13.49 nM T53381 C6I3MN 44420418 Ki = 309.03 nM T53381 CQV5N7 44420419 Ki = 436.52 nM T53381 CSQ5H2 44420423 Ki = 7.413 nM T53381 C1CFB6 44420428 Ki = 0.3981 nM T53381 CAW15U 44420431 Ki = 0.8318 nM T53381 C7C4QE 44426404 Ki = 13 nM T53381 CE3XQ2 44426405 Ki = 2.7 nM T53381 C21KYB 44428845 Ki = 1.549 nM T53381 C91BHJ 44428846 Ki = 3.631 nM T53381 CCLI02 44428847 Ki = 7.413 nM T53381 CE08JS 44428848 Ki = 2.344 nM T53381 CVH1Z5 44428849 Ki = 1.514 nM T53381 CY26IH 44428850 Ki = 26.92 nM T53381 CRN18J 44428851 Ki = 3.236 nM T53381 CBK87I 44431173 Ki = 30.2 nM T53381 CX3D0B 44431174 Ki = 0.3 nM T53381 C9HD0G 44431180 Ki = 0.2 nM T53381 CB3A8T 44431184 Ki = 0.5 nM T53381 C09VIB 44431192 Ki = 1.5 nM T53381 C43SCL 44431194 Ki = 0.8 nM T53381 C4G7QF 44431545 Ki = 5.2 nM T53381 C8OP5V 44431546 Ki = 3.2 nM T53381 C0B5TC 44431547 Ki = 2.4 nM T53381 CCXB24 44431548 Ki = 2.5 nM T53381 C5QI0V 44431551 Ki = 3.3 nM T53381 C2R4TP 44431553 Ki = 1.4 nM T53381 COIS42 44431554 Ki = 4.8 nM T53381 C0APQ4 44431555 Ki = 3.4 nM T53381 CJT34W 44431557 Ki = 2.1 nM T53381 CF76RP 44431560 Ki = 0.68 nM T53381 CY8C0V 44431562 Ki = 5.1 nM T53381 C2UD6M 44431564 Ki = 7 nM T53381 C4J0TG 44431574 Ki = 5 nM T53381 C0C8TU 44431587 Ki = 0.8 nM T53381 C1QV6S 44431590 Ki = 14 nM T53381 CF3ST7 44431594 Ki = 2.2 nM T53381 CA9O2E 44431599 Ki = 11 nM T53381 CX9YA2 44431602 Ki = 0.64 nM T53381 C9OSE8 44431607 Ki = 6.2 nM T53381 CT0LP1 44431611 Ki = 1.5 nM T53381 C46NHX 44431612 Ki = 15 nM T53381 C3IA4W 44431613 Ki = 64 nM T53381 C5QJ8S 44431614 Ki = 48 nM T53381 CXD1Q9 44431615 Ki = 44 nM T53381 C0WPS6 44431616 Ki = 3.6 nM T53381 C4SZA3 44431617 Ki = 5.5 nM T53381 CE6L0D 44431618 Ki = 9.4 nM T53381 CS9N3Q 44431620 Ki = 0.14 nM T53381 CEWQ41 44433348 Ki = 6.7 nM T53381 C64POV 44449245 EC50 = 336 nM T53381 CX7Z6I 44449247 EC50 > 10000 nM T53381 CO9NC7 44449248 EC50 > 10000 nM T53381 C1P3XZ 44449249 EC50 > 10000 nM T53381 CN9BI4 44449276 EC50 > 10000 nM T53381 CYM30S 44449277 EC50 > 10000 nM T53381 CS5WB3 44449278 EC50 > 10000 nM T53381 CH74NV 44449303 EC50 > 10000 nM T53381 C8VO6A 44449304 EC50 > 10000 nM T53381 CI4T2K 44449305 EC50 > 10000 nM T53381 C70SEG 44449306 EC50 > 10000 nM T53381 C0M7UN 44449337 EC50 > 10000 nM T53381 C4THN7 44449338 EC50 > 10000 nM T53381 C1O6QI 44449657 EC50 > 10000 nM T53381 C6QCN8 44449686 EC50 = 3190 nM T53381 CH5RL7 44449690 EC50 > 10000 nM T53381 CS3LB0 44449691 EC50 > 10000 nM T53381 CFL25O 44449692 EC50 = 1390 nM T53381 CSZB25 44449694 EC50 > 10000 nM T53381 CJ8WL7 44449723 EC50 > 10000 nM T53381 C8XHB5 44449724 EC50 > 10000 nM T53381 C6ZG3O 44449725 EC50 = 634 nM T53381 CMLE59 44449730 EC50 = 319 nM T53381 C12XGE 44456400 Ki > 10000 nM T53381 CGO23X 44460394 Ki > 5000 nM T53381 CLVD72 44460423 Ki = 170 nM T53381 C7T2KE 44460449 Ki > 5000 nM T53381 CVJ72X 44460477 Ki = 34.5 nM T53381 CT5M7N 44460522 Ki = 1107 nM T53381 CV3IW1 44461012 Ki = 894 nM T53381 C1PI3F 44462130 Ki = 2000 nM T53381 CB5MJ4 44469973 Ki = 0.66 nM T53381 CQ18ZE 44470113 Ki = 1.6 nM T53381 CJ10OZ 44531812 Ki = 1995 nM T53381 CAR23X 44568818 Ki = 125.89 nM T53381 CAO31F 44568917 Ki = 102.33 nM T53381 CE3GV8 44568918 Ki = 169.82 nM T53381 CVF30Y 44574044 EC50 > 10000 nM T53381 CCD72N 44574045 EC50 = 729 nM T53381 CMS20J 44574074 EC50 = 391 nM T53381 C92YUA 44574075 EC50 = 146 nM T53381 C9NU2C 44574076 EC50 > 3570 nM T53381 CX4Y0K 44574078 EC50 = 119 nM T53381 CU9X8G 44574079 EC50 = 656 nM T53381 CAT57X 44574103 EC50 > 10000 nM T53381 CXZ0J3 44574104 EC50 > 10000 nM T53381 CES4X0 44574105 EC50 > 10000 nM T53381 C62AYR 44574106 EC50 > 10000 nM T53381 CX98MY 44574107 EC50 > 3400 nM T53381 CDER54 44574132 EC50 > 10000 nM T53381 C4S2OQ 44574133 EC50 > 10000 nM T53381 C96NQZ 44574134 EC50 = 276 nM T53381 CKR69S 44574135 EC50 = 276 nM T53381 CL37FD 44574137 EC50 > 10000 nM T53381 CG0RM2 44574138 EC50 > 4100 nM T53381 CD87ZE 44574834 EC50 > 10000 nM T53381 C2YF8O 44574874 EC50 > 10000 nM T53381 CFQJ71 44574875 EC50 > 10000 nM T53381 CB1R3O 44574876 EC50 > 10000 nM T53381 CR8SF7 44574877 EC50 = 3500 nM T53381 CN94EW 44574878 EC50 > 10000 nM T53381 C8L6CN 44574934 EC50 > 10000 nM T53381 CVN8Z4 44574935 EC50 = 364 nM T53381 C9QAM5 44574936 EC50 > 10000 nM T53381 CV06SB 44574938 EC50 > 10000 nM T53381 C3QWO0 44574986 EC50 = 301 nM T53381 C4XHI5 44574989 EC50 > 10000 nM T53381 C9F6EB 44593557 EC50 > 7000 nM T53381 C51AJZ 44593577 EC50 > 10000 nM T53381 CDA54Q 44593580 EC50 > 10000 nM T53381 C1SN7Y 44593709 Ki = 4.571 nM T53381 CWO70X 45260703 Ki = 1202.26 nM T53381 C4VOW6 45260704 Ki = 223.87 nM T53381 CQ0R5Y 45264581 EC50 = 8.913 nM T53381 C39CDN 45264638 EC50 = 51.29 nM T53381 C0F4TJ 45268939 Ki = 0.1698 nM T53381 C05PBD 46176231 IC50 > 10000 nM T53381 C2L5UH 46182745 IC50 > 10000 nM T53381 C0ABR3 46846073 Ki = 331.13 nM T53381 C7ZEI6 46881382 Ki = 20.42 nM T53381 CN0Q2A 46881443 Ki = 57.54 nM T53381 CGX02N 46881444 Ki = 50.12 nM T53381 C4U6RH 46881493 Ki = 25.7 nM T53381 CV7R9S 46881494 Ki = 6.607 nM T53381 C24QFO 46882032 Ki > 1000 nM T53381 C3GQW6 46882033 Ki > 1000 nM T53381 CPG6U5 46882034 Ki = 6.31 nM T53381 CYB37P 46882085 Ki = 6.761 nM T53381 CD8CX3 46882086 Ki > 1000 nM T53381 C57GAO 46882087 Ki > 1000 nM T53381 CV3QW9 46882088 Ki = 354.81 nM T53381 C5ZDY3 46915370 Ki = 497 nM T53381 CI4XZ1 46934637 Ki = 1.479 nM T53381 CK1Z0M 46934639 Ki = 14.13 nM T53381 CU0TB9 46934641 Ki = 2.512 nM T53381 CR6JV7 46934643 Ki = 4.074 nM T53381 C14ZLO 46934645 Ki = 16.22 nM T53381 C2N9JZ 46934787 Ki = 39.81 nM T53381 CI4U0L 46934789 Ki = 8.511 nM T53381 C8HVG6 46934791 Ki = 32.36 nM T53381 CA51JI 46934793 Ki = 1.38 nM T53381 CB4Z7D 46934945 Ki = 4.786 nM T53381 C2LZJ0 49783209 Ki = 2276 nM T53381 C57SMG 49783415 Ki > 10000 nM T53381 C0TG6I 49783419 Ki > 10000 nM T53381 C0D5GI 49796077 Ki < 1000 nM T53381 C6ZRD7 49797187 Ki = 295.12 nM T53381 C63FGJ 49797190 Ki = 204.17 nM T53381 C2RY0J 50878551 Ki > 10000 nM T53381 C1W6TV 50898777 Ki > 10000 nM T53381 CXMZ73 50898778 Ki > 10000 nM T53381 C8EU7J 50905381 Ki = 0.2455 nM T53381 CW7FI3 50905585 Ki = 0.3236 nM T53381 CIL56G 50905588 Ki = 17.38 nM T53381 C5M6VO 50905589 Ki = 15.49 nM T53381 CE4KP1 51050257 Ki > 10000 nM T53381 CQG7X2 51349173 EC50 > 10000 nM T53381 CLW3B0 52940951 Ki = 0.7413 nM T53381 CWYS78 52941004 Ki = 3.715 nM T53381 CE0X9W 52941056 Ki = 17.78 nM T53381 C40WVE 52941624 Ki = 3.981 nM T53381 CV7HZ6 52942047 Ki = 13.49 nM T53381 C5Y3VS 52942152 Ki = 0.5129 nM T53381 CO9J6M 52943356 Ki = 0.912 nM T53381 CRL3P0 52944615 Ki = 7.079 nM T53381 C4N6ET 52944674 Ki = 15.14 nM T53381 CDQ27E 52945156 Ki = 2.754 nM T53381 CPI9F4 52945803 Ki = 0.389 nM T53381 CGZ1R7 52947088 Ki = 14.13 nM T53381 CNH57S 52947579 Ki = 0.1778 nM T53381 CX04NC 52948119 Ki = 5.248 nM T53381 C9YBJ3 52948823 Ki = 1.202 nM T53381 CCQZ15 52949448 Ki = 0.8128 nM T53381 CGY45S 53248361 Ki = 98 nM T53381 CE9L8G 53248365 Ki = 181 nM T53381 C4H5JI 53327748 Ki = 1.995 nM T53381 C1YX4A 53327991 Ki = 0.5012 nM T53381 CUP50Y 53327992 Ki = 5.012 nM T53381 CZ1B6D 53328115 Ki = 1318.26 nM T53381 CT0D9O 53328116 Ki = 630.96 nM T53381 CGB3U6 53328311 Ki = 45.71 nM T53381 CIWJ61 53328312 Ki = 43.65 nM T53381 CW36HN 53328313 Ki = 389.05 nM T53381 C6NUW4 53328314 Ki = 33.88 nM T53381 C7XCQ4 53328315 Ki = 38.9 nM T53381 CJ7TY9 53328316 Ki = 30.9 nM T53381 C76NJW 53328503 Ki = 691.83 nM T53381 CB1D8L 53328504 Ki = 1513.56 nM T53381 CY9JI7 53328505 Ki = 69.18 nM T53381 C5FHA1 53328506 Ki = 63.1 nM T53381 CCM7S9 53328507 Ki = 72.44 nM T53381 C7YN2M 53328508 Ki = 67.61 nM T53381 CD7EB0 53328684 Ki = 53.7 nM T53381 CQGE30 53328685 Ki = 51.29 nM T53381 CNSU94 53328686 Ki = 97.72 nM T53381 CY51RC 53328687 Ki = 77.62 nM T53381 C9L0ZI 53328872 Ki = 912.01 nM T53381 C67YNQ 53328873 Ki = 75.86 nM T53381 CMOZ61 53475319 Ki = 1184 nM T53381 CGX1W2 53779053 Ki = 193 nM T53381 C6W1RA 56649648 Ki = 27 nM T53381 C2SW7J 56649649 Ki = 73 nM T53381 CQTR49 56649650 Ki = 19 nM T53381 CA6B2I 56668277 Ki = 620 nM T53381 CCW38Z 56945164 Ki = 5.754 nM T53381 CN6XE8 56945165 Ki = 67.61 nM T53381 CPE6C7 56945166 Ki = 93.33 nM T53381 C4L7GW 56945167 Ki = 67.61 nM T53381 CL68PZ 56946472 Ki = 31.62 nM T53381 CJ98DO 56946474 Ki = 6.31 nM T53381 CB8J2F 56946573 Ki = 3.89 nM T53381 CCBY53 56946575 Ki = 389.05 nM T53381 CMO0U3 56946577 Ki = 141.25 nM T53381 CJZ3P4 56946579 Ki = 154.88 nM T53381 CXUW26 56961460 IC50 < 5 nM T53381 CX74AS 56961506 IC50 < 5 nM T53381 C9WP3O 56961507 Ki = 20.7 nM T53381 C1TC7Q 56963799 Ki > 10000 nM T53381 C53OMP 57391554 IC50 = 100 nM T53381 CDTG05 57393527 Ki = 0.8128 nM T53381 CYZD14 57395043 IC50 = 501.19 nM T53381 C2CEB9 57398562 IC50 = 31.62 nM T53381 C1NGZ7 57400229 IC50 = 25.12 nM T53381 C3TYE1 57401435 IC50 = 398.11 nM T53381 CM7EN2 57401436 IC50 = 79.43 nM T53381 C8EFT7 57402251 Ki > 1000 nM T53381 C4AHC0 57929587 Ki = 3.7 nM T53381 C6LQ7C 57929588 Ki = 9.4 nM T53381 CWF57Q 57929612 Ki = 4.8 nM T53381 CI64JE 58149995 Ki = 15 nM T53381 C41YWP 58150016 Ki = 3.4 nM T53381 CXE03T 59151542 Ki = 16 nM T53381 C3GT1H 59151543 Ki = 23 nM T53381 C9D4KG 59151549 Ki = 160 nM T53381 CTI2Q0 59151563 Ki = 8.7 nM T53381 C7T2XI 59151572 Ki = 250 nM T53381 C5XT8Q 59151583 Ki = 7.5 nM T53381 CM0UZ4 59151610 Ki = 39 nM T53381 C0TA6I 59151612 Ki = 820 nM T53381 CMPQ30 59151614 Ki = 26 nM T53381 CJ5R1B 59151621 Ki = 8.5 nM T53381 C8IAO2 59151651 Ki = 54 nM T53381 CZ1FX8 59151668 Ki = 420 nM T53381 CST67R 59151671 Ki = 11 nM T53381 C1SBP9 69781970 Ki = 3.981 nM T53381 CCD2L1 69782867 Ki = 0.389 nM T53381 C6SN2P 71449516 Ki = 323.59 nM T53381 CFS69A 71450901 Ki = 25.12 nM T53381 C75EQJ 71452768 Ki = 92 nM T53381 C31VFN 71454865 Ki = 8.913 nM T53381 CORB94 71458492 Ki = 3.981 nM T53381 CA6NI7 71462043 Ki = 0.7079 nM T53381 CD9G8B 71521478 Ki = 724.44 nM T53381 CSV0G5 71521479 Ki = 25.12 nM T53381 CGN2M7 71521480 Ki = 83.18 nM T53381 CDS15J 71659980 Ki = 1.514 nM T53381 CH6J4G 71817545 Ki = 630.96 nM T53381 CH54DW 71817546 Ki = 2.239 nM T53381 C3NO8R 71817548 Ki = 12.88 nM T53381 CRTD80 71817857 Ki = 1348.96 nM T53381 CBTX18 71817858 Ki = 18.2 nM T53381 CRYP87 71817860 Ki = 83.18 nM T53381 CC65OA 73213195 Ki > 10000 nM T53381 CW83DK 73213196 Ki = 293 nM T53381 CCV91B 73346042 Ki = 62.6 nM T53381 CX01MD 73349178 Ki = 18.2 nM T53381 CBW1D8 73356785 Ki = 1.905 nM T53381 C8IDL3 75306277 Ki = 794.33 nM T53381 CFN6P8 76071738 IC50 > 10000 nM T53381 CW61JI 76071739 IC50 = 250.7 nM T53381 C04HNK 76308473 Ki = 3.631 nM T53381 C8M3OX 76323009 Ki = 4.786 nM T53381 COT51G 76326561 Ki = 7.413 nM T53381 CFV87U 76330228 Ki = 1.549 nM T53381 C3Z1TP 78815633 Ki = 1.349 nM T53381 CL9AI7 85469698 IC50 = 1758 nM T53381 CGO74F 85469753 IC50 = 7426 nM T53381 C91LTS 85469754 IC50 = 10.07 nM T53381 CS9DG8 85469755 IC50 = 493.3 nM T53381 CU6R1L 85469756 IC50 = 1862 nM T53381 CTRN10 85469757 IC50 = 957.2 nM T53381 CU3P0H 85469808 IC50 = 115.5 nM T53381 C74PRV 85469809 IC50 = 866.4 nM T53381 CUOH37 85469811 IC50 = 36.62 nM T53381 CKNG20 85469812 IC50 = 239.9 nM T53381 C6-MAR-04 85469868 IC50 = 63.54 nM T53381 CJQ9O7 85469869 IC50 = 11.31 nM T53381 C4HA3I 85469870 IC50 = 80550 nM T53381 C9NL2S 85469871 IC50 = 10630 nM T53381 C1J0GW 85469872 IC50 = 35.16 nM T53381 CVM3B2 85469873 IC50 = 163.7 nM T53381 CYI5J6 85469930 IC50 = 31.28 nM T53381 CZI3Y2 85469931 IC50 = 12.87 nM T53381 CAS6Y8 85469932 IC50 = 1235 nM T53381 C7PXK3 85469933 IC50 = 343.6 nM T53381 C7XI0F 85469934 IC50 = 122 nM T53381 CLBA19 86344174 IC50 = 474.3 nM T53381 CL9GY7 90645592 Ki = 0.5754 nM T53381 CI49HV 90645593 Ki = 0.912 nM T53381 C41AGZ 90645594 Ki = 3.236 nM T53381 C1L0PW 90645595 Ki = 1.175 nM T53381 C7JL5G 90645596 Ki = 0.3715 nM T53381 C89TJI 90645597 Ki = 0.1413 nM T53381 CHBC38 90645598 Ki = 0.05623 nM T53381 C4MLA7 90645599 Ki = 1 nM T53381 C0WXR7 90645600 Ki = 4.074 nM T53381 CN8TF6 90645601 Ki = 1.66 nM T53381 CKN56Z 90645602 Ki = 5.012 nM T53381 CYQ3M8 90645603 Ki = 3.311 nM T53381 C45MSD 90645604 Ki = 5.495 nM T53381 C4I6EW 90645605 Ki = 0.7586 nM T53381 CH92LD 90645606 Ki = 2.291 nM T53381 C7YQM3 101333429 Ki = 426 nM T53381 CE0ZC6 101876962 Ki = 478.63 nM T53381 CJ15CM 102012413 Ki = 253122 nM T53381 CA43MY 117839022 IC50 = 1107 nM T53381 CWR6I1 118112300 IC50 = 8000 nM T53381 CI7NQ9 118716698 Ki = 14.79 nM T53381 CGO9W4 118716699 Ki = 25.12 nM T53381 CVDI36 118716700 Ki = 4.677 nM T53381 C94AFL 118716701 Ki = 42.66 nM T53381 CTX92K 118716702 Ki = 51.29 nM T53381 CG02WP 118716703 Ki = 37.15 nM T53381 CTNL85 118716704 Ki = 8.128 nM T53381 CM1Y8W 118716705 Ki = 22.91 nM T53381 C42MOT 118716706 Ki = 20.42 nM T53381 C78ARU 118716707 Ki = 10.96 nM T53381 CO5TG3 118716708 Ki = 28.18 nM T53381 CNF78L 118716709 Ki = 39.81 nM T53381 C9CB1Q 118716710 Ki = 26.92 nM T53381 C3F6EQ 118716711 Ki = 89.13 nM T53381 C0L6YO 118716712 Ki = 416.87 nM T53381 CX2AC4 118716713 Ki = 12.3 nM T53381 CL1EU8 118716714 Ki = 10.72 nM T53381 C0V7GJ 118716715 Ki = 7.079 nM T53381 CRBI65 118716716 Ki = 26.3 nM T53381 C70IPZ 118716717 Ki = 5.754 nM T53381 CBI30N 118716718 Ki = 0.912 nM T53381 C7UBN8 118716719 Ki = 9.772 nM T53381 CV8HA2 118716720 Ki = 23.44 nM T53381 C30ZJB 118716721 Ki = 13.18 nM T53381 C58MND 118716722 Ki = 19.05 nM T53381 CO6T4G 118716723 Ki = 35.48 nM T53381 C8RVX4 118717455 Ki = 489.78 nM T53381 C5IM1N 118717456 Ki = 204 nM T53381 CBCU90 118717457 Ki = 213.8 nM T53381 CN4LJ2 118717458 Ki = 478.63 nM T53381 CZ35PU 118717459 Ki = 371.54 nM T53381 C9BP7A 118717460 Ki = 489.78 nM T53381 CFCM61 118717461 Ki = 229 nM T53381 C8C6ZW 118717462 Ki = 758.58 nM T53381 CR8Z0F 118718431 Ki = 1100 nM T53381 CUEG14 122179430 Ki = 0.4 nM T53381 CV51WL 122179431 Ki = 27.5 nM T53381 C5PW9Y 123141715 IC50 = 31.6 nM T53381 C03AHG 123183757 IC50 = 49.6 nM T53381 CK4ZO0 123183788 IC50 = 60.6 nM T53381 C17PEO 123204312 IC50 = 1621 nM T53381 C9W8OX 123311113 IC50 = 3464 nM T53381 CCK90I 123322716 IC50 = 457.5 nM T53381 C8AKN7 123368349 IC50 = 274 nM T53381 C5I2VU 123378354 IC50 = 436.2 nM T53381 C9ZCI2 123387804 IC50 = 0.4 nM T53381 C6LRF9 123393714 IC50 = 996.1 nM T53381 CU7CX9 123415538 IC50 = 21.7 nM T53381 C3HJV5 123437117 IC50 = 196.8 nM T53381 CO3CT2 123472560 IC50 = 1345 nM T53381 C8RU2P 123475619 IC50 = 162.2 nM T53381 C8XV2H 123562321 IC50 = 0.4 nM T53381 CF2R5U 123576734 IC50 = 883.2 nM T53381 C1HE3L 123644751 IC50 = 410.2 nM T53381 C9IR4A 123667086 IC50 = 0.3 nM T53381 C3CK5L 123688273 IC50 = 143.9 nM T53381 CAN97K 123752717 IC50 = 1554 nM T53381 C9CO7R 123801568 IC50 = 5208 nM T53381 CI4TU7 123854385 IC50 = 94 nM T53381 C2T0KW 123986550 IC50 = 3794 nM T53381 C7T0GE 124018870 IC50 = 0.4 nM T53381 CM57GR 126720252 Ki = 1270 nM T53381 CTBN56 127026052 Ki < 10000 nM T53381 CQ0ZT9 127035062 Ki = 467 nM T53381 CU49VE 127036186 Ki < 10000 nM T53381 CG06BD 127036932 Ki = 1318.26 nM T53381 CVW71O 127036953 Ki = 1122.02 nM T53381 CXR71M 127038002 Ki = 0.5129 nM T53381 CL5N3P 127038713 Ki = 10.47 nM T53381 C89SOL 127040060 Ki = 14.45 nM T53381 CQ3L8Z 127040156 Ki = 22.91 nM T53381 CCH14Q 127041710 IC50 = 16.73 nM T53381 C8A1TO 127043026 IC50 = 3717 nM T53381 C3GX2A 127044893 IC50 = 37.4 nM T53381 C6P4LV 127044894 IC50 = 15.8 nM T53381 C70SOF 127044906 IC50 = 457.1 nM T53381 C1I6UZ 127044911 IC50 = 0.4 nM T53381 CX9PE0 127044912 IC50 = 0.1 nM T53381 CXKQ86 127044916 IC50 = 10.6 nM T53381 CL40YC 127045050 IC50 = 1.7 nM T53381 C3ARM8 127046608 Ki = 880 nM T53381 CNM5P2 127046693 Ki = 130 nM T53381 C37WYI 127046694 Ki = 65 nM T53381 CI10VG 127046766 Ki > 940 nM T53381 C5BU9Z 127047696 Ki > 940 nM T53381 CN2KE8 131978695 IC50 = 640.6 nM T53381 CGHO19 132060770 Ki = 3524 nM T53381 CT81OY 132060776 Ki = 1767 nM T53381 CFXL21 132060812 Ki = 2738 nM T53381 CAVB41 132584404 Ki > 10000 nM T53381 C6D1HC 134132279 Ki = 1778.28 nM T53381 CM4XE8 134133829 Ki = 32.36 nM T53381 CKH7W6 134137025 Ki = 38.9 nM T53381 C5A6XO 134138438 Ki = 100 nM T53381 CP67BZ 134138882 IC50 > 10000 nM T53381 CB0S8Y 134139869 Ki = 1.349 nM T53381 CYW9L4 134142282 IC50 = 4038 nM T53381 C46ZTY 134143085 Ki = 123.03 nM T53381 C7GT5Y 134145079 IC50 > 10000 nM T53381 CXN73G 134147055 Ki = 1.318 nM T53381 C1QZ5S 134147190 IC50 = 1456 nM T53381 CS2OC5 134147929 Ki = 2.57 nM T53381 CBU81N 134149168 Ki > 10000 nM T53381 C7HT1Z 134149596 Ki = 1.738 nM T53381 C0CEH2 134149598 IC50 = 8392 nM T53381 CEU53H 134149777 Ki = 34.67 nM T53381 C4BH9V 134150497 Ki = 4.571 nM T53381 CF46WD 134150827 IC50 > 10000 nM T53381 C9IAC0 134152568 Ki = 3.09 nM T53381 CDWP64 134153527 Ki = 213.8 nM T53381 C6S0VM 134157330 Ki = 95.5 nM T53381 CBL29F 134157566 IC50 > 10000 nM T53381 C25RED 137631359 Ki = 6.607 nM T53381 C19JKQ 137638321 Ki = 5.012 nM T53381 CA03VC 137639125 Ki = 79.43 nM T53381 CZ4TA9 137640201 Ki = 302 nM T53381 CE8N4S 137641762 Ki > 10000 nM T53381 CU1O2P 137642386 Ki = 5.495 nM T53381 CKS5V0 137643541 Ki > 10000 nM T53381 C96EAP 137646245 Ki = 77.62 nM T53381 CW2L7Z 137651819 Ki = 5.888 nM T53381 CR9F3Q 137653203 Ki > 10000 nM T53381 CMDV74 144096985 Ki = 9.1 nM T53381 CN67YQ 144096995 Ki = 8.6 nM T53381 C91RQY 145949210 Ki = 33.88 nM T53381 CL0XY8 145950240 Ki = 48.98 nM T53381 C45LBY 145951352 Ki = 37.15 nM T53381 CB3O4C 145951457 Ki = 102.33 nM T53381 CE3ZM8 145953314 Ki = 3.715 nM T53381 C6VO0S 145955016 Ki > 1000 nM T53381 CT9I0G 145956955 Ki = 0.3311 nM T53381 C75KTN 145958538 Ki = 28.18 nM T53381 CX56QA 145960918 Ki = 6.166 nM T53381 CFBX59 145962085 Ki = 295.12 nM T53381 C2FNR9 145962342 Ki = 0.0631 nM T53381 CE9I6G 145962368 Ki = 5.129 nM T53381 C0G7JA 145962478 Ki = 2.138 nM T53381 C3DGE5 145962817 Ki = 104.71 nM T53381 C2HL4E 145962945 Ki = 2.239 nM T53381 C7BC0I 145963755 Ki = 13.18 nM T53381 C64TUP 145963761 Ki = 17 nM T53381 CQU59F 145963832 Ki > 94 nM T53381 CO6G4Y 145964722 Ki = 170 nM T53381 CN4K5B 145965240 Ki = 86 nM T53381 CZ86PI 145965488 Ki = 62 nM T53381 C0TU9I 145965623 Ki = 1.1 nM T53381 CT5E6B 145966751 Ki = 1.5 nM T53381 CVH7O4 145967266 Ki = 310 nM T53381 CZSN84 145967270 Ki = 4.3 nM T53381 CIN42D 145967562 Ki = 12 nM T53381 C8AOB7 145967761 Ki = 9.5 nM T53381 CBPU13 145968055 IC50 = 102.85 nM T53381 CTJ0X5 145968736 IC50 = 826.47 nM T53381 CTP81Y 145968741 IC50 = 736.47 nM T53381 C9M7ZG 145969396 Ki = 65 nM T53381 CT9FQ7 145969986 IC50 = 452.84 nM T53381 CDLX87 145970204 IC50 = 287.18 nM T53381 C7IGH9 145970995 Ki = 0.85 nM T53381 CL3D9C 145972633 Ki = 17 nM T53381 CGVL80 145974123 Ki = 38 nM T53381 CQIB05 145975238 Ki = 0.3 nM T53381 CF8ET9 145975365 Ki > 94 nM T53381 C0W3YR 145977627 Ki = 3.9 nM T53381 C6P3SR 153287553 Ki = 1000 nM T53381 CV9G7Z 153287572 Ki > 10000 nM T53381 CO85KL 153287574 Ki > 10000 nM T53381 C7N0VH 155512508 Ki > 1000 nM T53381 C7W1OH 155513940 Ki = 5.888 nM T53381 CV8F7A 155515301 Ki = 89.13 nM T53381 CT4U8D 155517137 Ki = 316.23 nM T53381 CAV5Y1 155519565 Ki > 1000 nM T53381 CUSA24 155519891 Ki > 10000 nM T53381 CL07FB 155521817 Ki = 53.7 nM T53381 CXEB36 155523275 Ki = 95.5 nM T53381 CYZ60F 155524736 Ki = 190.55 nM T53381 CD5BI1 155525649 Ki = 87.1 nM T53381 C8GC1P 155526628 Ki = 5.754 nM T53381 CIO6V1 155528183 Ki > 1000 nM T53381 C7FR8Y 155529117 Ki = 29.51 nM T53381 CF2DM6 155529314 Ki = 1.202 nM T53381 C3ZL2V 155531279 Ki = 125.89 nM T53381 C3R4YM 155532148 Ki = 1.738 nM T53381 C3MXL6 155532834 Ki = 1.023 nM T53381 CTU64O 155533099 Ki = 10 nM T53381 CU3YE7 155534933 Ki = 69.18 nM T53381 CB79ZW 155536080 Ki > 10000 nM T53381 CQG68A 155536202 Ki = 75.86 nM T53381 CFH7K5 155542074 Ki = 30.2 nM T53381 C91VXF 155544397 Ki > 1000 nM T53381 CR54LA 155544513 Ki = 4.365 nM T53381 CXH9A8 155549493 Ki > 1000 nM T53381 C9XQ8H 155552820 Ki = 177.83 nM T53381 C4LOH3 155555858 Ki = 15.85 nM T53381 C0CV6O 155557695 Ki = 57.54 nM T53381 C3UCM2 155557792 Ki = 7.413 nM T53381 C20QMI 155558704 Ki > 1000 nM T53381 CE0HN5 155559841 Ki > 1000 nM T53381 C8ZKT3 155562124 Ki = 5.012 nM T53381 C71MOD 155563001 Ki = 7.079 nM T53381 C3DK0P 155565218 Ki = 95.5 nM T53381 CVU9O2 155565448 Ki = 16.6 nM T53381 C19PZX 155565707 Ki > 1000 nM T53381 CRX52O 155567200 Ki = 25.12 nM T53381 D00GEE 92766 Ki = 253 nM T53381 D01BJZ 9817640 Ki = 158.49 nM T53381 D02NNS 9845181 Ki = 1.3 nM T53381 D05ZUX 44207909 Ki >= 1000 nM T53381 D06QKW 2765 EC50 = 125.89 nM T53381 D06UBB 123981 Ki = 126 nM T53381 D07QCC 10946567 Ki = 1.2 nM T53381 D08XTL 9866614 Ki = 80 nM T53381 D09ZUW 6603904 Ki = 34 nM T53381 D0BI4T 53315878 Ki = 4500 nM T53381 D0D8GV 9830741 Ki = 122 nM T53381 D0DP8I 132266 Ki = 0.1698 nM T53381 D0EO4F 9891167 Ki = 0.312 nM T53381 D0H3CW 9839317 Ki = 72 nM T53381 D0L5MW 181743 Ki = 340 nM T53381 D0N7UE 10198248 Ki = 12302.69 nM T53381 D0O3GF 1220 Ki > 1000 nM T53381 D0O6MG 3567002 Ki = 12.59 nM T53381 D0Q4PY 9888164 Ki = 505 nM T53381 D0Q7ZR 9890547 Ki = 0.252 nM T53381 D0T2RY 9948320 Ki = 40 nM T53381 D0V6DJ 5640 Ki = 10 nM T53381 D0YZ3E 44435200 Ki = 4100 nM T53381 D0Z7EA 643606 Ki = 3.5 nM T53381 D0Z8OD 9887378 Ki = 372 nM T65879 D0E3TC 44259 IC50 = 233 nM T65879 D0Z5DM 5081913 IC50 > 100000 nM T65879 D03BNU 59604787 IC50 > 10000 nM T65879 D01OLO 9820526 IC50 = 1300 nM T65879 C2XU5O 162883 IC50 = 600 nM T65879 CAS18T 359052 IC50 = 21000 nM T65879 CYN49L 575802 IC50 > 100000 nM T65879 CU73ST 599501 IC50 > 100000 nM T65879 CL5E6W 607775 IC50 = 4000 nM T65879 CR98MZ 613528 IC50 = 2800 nM T65879 C0ZI1F 2756534 IC50 > 30000 nM T65879 CT6P3F 2782903 IC50 = 24000 nM T65879 CMC16L 2782960 IC50 > 100000 nM T65879 C2DQY6 5324413 Ki > 30000 nM T65879 C04EDX 9549298 IC50 = 200 nM T65879 CGH0R4 9796523 IC50 = 420 nM T65879 CD71UI 9813758 IC50 = 4000 nM T65879 C6TZ7U 9813880 IC50 = 990 nM T65879 CM5Z8X 9869943 IC50 = 50000 nM T65879 C6MZB1 9900652 IC50 = 1600 nM T65879 C3QW5M 9922100 IC50 = 870 nM T65879 C6PW4K 9989716 Ki > 30000 nM T65879 CW59RK 10109125 IC50 = 1700 nM T65879 C9ARB8 10126159 IC50 = 12100 nM T65879 CU4F6P 10215156 IC50 = 400 nM T65879 CSGD16 10246246 IC50 = 90 nM T65879 CF9MV3 10410982 IC50 = 6918 nM T65879 C4JZ7U 10448840 IC50 = 300 nM T65879 CLB09P 11075446 IC50 = 200 nM T65879 C4ZV5I 11149107 IC50 = 15848.93 nM T65879 CRP61Y 11156148 IC50 = 7943.28 nM T65879 CJ7U4I 11161778 IC50 = 270 nM T65879 C9LA7N 11164332 IC50 = 4000 nM T65879 CNCT02 11173949 IC50 = 3500 nM T65879 CW5C9X 11186250 IC50 = 1584.89 nM T65879 C9GY2P 11207091 IC50 = 10000 nM T65879 CT19ID 11207978 IC50 = 6309.57 nM T65879 C35AIB 11287153 IC50 = 600 nM T65879 CBOP58 11293798 Ki > 10000 nM T65879 C9TOG5 11304835 IC50 = 3162.28 nM T65879 C9CWY7 11323357 IC50 = 3981.07 nM T65879 CV43QF 11336440 IC50 = 3981.07 nM T65879 CM0GX5 11350427 IC50 = 1995.26 nM T65879 C26BZX 11362471 Ki > 10000 nM T65879 CWXB93 11397177 Ki > 10000 nM T65879 CU76FI 11402873 IC50 = 15848.93 nM T65879 CVX70O 11427162 IC50 = 10000 nM T65879 C8VT9G 11436911 IC50 = 10000 nM T65879 C7X4HG 11448486 IC50 = 2600 nM T65879 CM21YJ 11453049 IC50 = 1995.26 nM T65879 CTG83F 11539329 Ki > 1500 nM T65879 CMIL86 11590363 Ki > 1500 nM T65879 CH7P9Z 11608743 IC50 > 30000 nM T65879 CGX96V 11626927 IC50 < 15848.93 nM T65879 C9T6SC 11640926 Ki > 1500 nM T65879 CJ9KN7 11683817 IC50 > 10000 nM T65879 CU0E8O 11690457 Ki > 2000 nM T65879 CB0AP2 11705863 Ki > 10000 nM T65879 C45EWD 11723489 IC50 = 3400 nM T65879 CZTR57 11954411 IC50 = 40 nM T65879 CG7X9F 12330558 IC50 > 100000 nM T65879 C93RGU 13441298 IC50 = 2000 nM T65879 C3QKT4 14355186 Ki = 4000 nM T65879 CEL3V6 14929458 IC50 = 1100 nM T65879 C3YRU7 15295578 IC50 > 50000 nM T65879 C2DKR4 15979284 IC50 = 398.11 nM T65879 CFPW41 16007116 Ki > 3800 nM T65879 C9TU1O 16046126 IC50 > 1000 nM T65879 CPJ94T 16047031 IC50 = 1995.26 nM T65879 C1Y0VG 16047033 IC50 = 5011.87 nM T65879 C1MA4Q 16047147 IC50 = 1995.26 nM T65879 CAPR-79 16047856 IC50 = 501.19 nM T65879 CJI9Z4 16047968 IC50 = 79.43 nM T65879 C2J6PS 16048084 IC50 = 2511.89 nM T65879 C6N5YF 16048085 IC50 = 1000 nM T65879 CM21OB 16048194 IC50 = 12589.25 nM T65879 CYQO76 16048303 IC50 = 5011.87 nM T65879 CTI58R 16048308 IC50 = 6309.57 nM T65879 C1QJ3P 16048414 IC50 = 7943.28 nM T65879 C6EU9X 16048415 IC50 = 3162.28 nM T65879 C2W0CV 16048543 IC50 = 10000 nM T65879 CL1NQ5 16048544 IC50 > 15848.93 nM T65879 CB8H0X 16663529 IC50 = 230 nM T65879 CF0H3L 17229016 IC50 = 89700 nM T65879 CT7OC2 20767724 IC50 = 670 nM T65879 C0T2VF 20823920 IC50 = 7830 nM T65879 CX0E5L 20823952 IC50 > 30000 nM T65879 CKQV75 20823956 IC50 = 14400 nM T65879 C9CUN2 20823959 IC50 = 6500 nM T65879 CD1K8E 20823960 IC50 = 1090 nM T65879 C1FE5V 20823975 IC50 = 3130 nM T65879 CG4H7B 20823982 IC50 = 1170 nM T65879 C9W2GS 20823986 IC50 = 7030 nM T65879 CKTI83 20823993 IC50 = 3480 nM T65879 C6A3PV 20823995 IC50 > 25000 nM T65879 CO27KL 20823998 IC50 > 100000 nM T65879 C2S7RG 20824041 IC50 = 4120 nM T65879 C9O4WF 20824060 IC50 = 1990 nM T65879 CXG6R2 21083789 IC50 > 20000 nM T65879 CS1MB4 21083790 IC50 = 3100 nM T65879 C7NMQ8 21083887 IC50 = 430 nM T65879 CP14LT 21083893 IC50 = 3500 nM T65879 CYC65I 21083894 IC50 = 4200 nM T65879 CA61QF 21083895 IC50 = 1900 nM T65879 C8WUE9 21083896 IC50 = 1000 nM T65879 CE20HN 21083898 IC50 = 6100 nM T65879 CWIR51 21083902 IC50 = 7600 nM T65879 CWTV36 21083906 IC50 = 3400 nM T65879 C9YMR6 21083908 IC50 = 20000 nM T65879 CULX07 21362669 IC50 = 1100 nM T65879 CU8J9B 21362674 IC50 = 700 nM T65879 C0FT4V 21362687 IC50 = 3000 nM T65879 CZ9TY2 21362689 IC50 = 1000 nM T65879 CT04LF 21362696 IC50 = 80 nM T65879 CF2O6I 21362697 IC50 = 3000 nM T65879 CLHK23 21362698 IC50 = 11000 nM T65879 CH48GT 21362699 IC50 = 3200 nM T65879 CMO14U 21362701 IC50 = 1300 nM T65879 CXE7L1 21362727 IC50 = 140 nM T65879 C7AWQ3 21362732 IC50 = 600 nM T65879 C8X9CQ 21362735 IC50 = 1800 nM T65879 C5E3VT 21362736 IC50 = 1800 nM T65879 COC1D6 21362741 IC50 = 170 nM T65879 CO8ZE5 21362748 IC50 = 1300 nM T65879 CE4V1D 21362749 IC50 = 600 nM T65879 CRDJ20 21362754 IC50 = 700 nM T65879 C1HT6L 21362756 IC50 = 8300 nM T65879 C40AEJ 22285027 IC50 = 390 nM T65879 CEXB18 22291652 IC50 = 14000 nM T65879 C5JH1P 22477600 IC50 = 3981.07 nM T65879 C6JV7W 23400934 IC50 = 13300 nM T65879 CD5S7O 23401001 IC50 = 11200 nM T65879 CC21PY 23648887 IC50 = 794.33 nM T65879 CMD65I 23648890 IC50 = 251.19 nM T65879 C4C2XA 23648920 IC50 = 1258.93 nM T65879 CWX53C 23648921 IC50 = 158.49 nM T65879 C2R1QH 23648953 IC50 = 50.12 nM T65879 CBA39U 23657350 IC50 = 390 nM T65879 CJM4C7 24219848 IC50 > 100000 nM T65879 C2UOE0 24766030 IC50 > 50000 nM T65879 CQN3Z7 24825710 IC50 = 4960 nM T65879 CI5B6S 24825779 IC50 > 50000 nM T65879 C8OUR0 24856835 IC50 = 398.11 nM T65879 C6CVK4 24959046 IC50 > 100000 nM T65879 CWE0L7 24983829 IC50 = 125.89 nM T65879 C2O0QA 24984297 IC50 = 199.53 nM T65879 CH32GJ 24984615 IC50 = 7943.28 nM T65879 C5RY8D 24984616 IC50 = 3981.07 nM T65879 C90YFT 24984774 IC50 = 316.23 nM T65879 CM3EI4 24984940 IC50 = 794.33 nM T65879 CQ2Z7T 24985115 IC50 = 199.53 nM T65879 C8O0JE 24985283 IC50 = 158.49 nM T65879 C90QPI 25093427 IC50 = 1110 nM T65879 CHTR48 25093428 IC50 = 940 nM T65879 CTD7L0 25093430 IC50 = 1260 nM T65879 CSX0O1 25093431 IC50 = 1450 nM T65879 C9AIZ8 25093432 IC50 = 1240 nM T65879 C2S5GF 25093433 IC50 = 2570 nM T65879 CQEP18 25093434 IC50 = 2930 nM T65879 CMJ8E0 25093435 IC50 = 13000 nM T65879 CW92XG 25093436 IC50 = 690 nM T65879 C8CJQ9 25093437 IC50 = 2800 nM T65879 CXM5Q4 25093438 IC50 = 4400 nM T65879 C9Y3PO 25093439 IC50 = 450 nM T65879 CNE20C 25093440 IC50 = 2330 nM T65879 C48WIP 25093441 IC50 = 910 nM T65879 CJL3O1 25093442 IC50 = 7990 nM T65879 CH27WL 25093443 IC50 = 220 nM T65879 C6FEC5 25093444 IC50 = 770 nM T65879 CN52FS 25093445 IC50 = 260 nM T65879 CU5CK2 25093446 IC50 = 170 nM T65879 C2YXB7 25093447 IC50 = 510 nM T65879 C6KFE7 25093448 IC50 = 650 nM T65879 COC9K8 25093449 IC50 = 820 nM T65879 C0N9GE 25093450 IC50 = 130 nM T65879 CR81QD 25093451 IC50 = 440 nM T65879 CRX17M 25093452 IC50 = 1080 nM T65879 CS1MO6 25093453 IC50 = 680 nM T65879 CT41VL 25093454 IC50 = 1340 nM T65879 CYC24O 25093455 IC50 = 1210 nM T65879 CU45OM 25093456 IC50 = 1260 nM T65879 C52VZG 25093457 IC50 = 190 nM T65879 CO58WP 25093458 IC50 = 260 nM T65879 C6P0DN 25093459 IC50 = 330 nM T65879 CD7WE8 25093460 IC50 = 1010 nM T65879 C6Q1ST 25169524 IC50 = 5000 nM T65879 C4D3FJ 25190920 IC50 > 15848.93 nM T65879 C1LZ2V 25190921 IC50 > 15848.93 nM T65879 CY9GT4 25190922 IC50 > 15848.93 nM T65879 CQMR47 25190923 IC50 > 15848.93 nM T65879 C5M8HZ 25190924 IC50 > 15848.93 nM T65879 CE8X6M 25190925 IC50 > 15848.93 nM T65879 CF6Z9S 25190926 IC50 > 15848.93 nM T65879 CUZ2N7 25190927 IC50 > 15848.93 nM T65879 CLFM35 25206064 IC50 > 50000 nM T65879 C56VHY 25219675 IC50 > 100000 nM T65879 CT9IN1 25263282 IC50 = 990 nM T65879 CN5E0F 25263283 IC50 = 4300 nM T65879 CW18IA 25263284 IC50 = 3400 nM T65879 CXN0J8 25263287 IC50 = 8100 nM T65879 C37JSG 25263288 IC50 = 840 nM T65879 CI7PA9 25263289 IC50 = 1100 nM T65879 CPC7D9 25263292 IC50 = 5000 nM T65879 CB7M1Z 25263293 IC50 = 8600 nM T65879 CNH56T 25263294 IC50 = 8300 nM T65879 C1Z6QP 25263295 IC50 = 1400 nM T65879 C02XNR 25263296 IC50 = 10000 nM T65879 CM0EF4 42618139 IC50 = 7943.28 nM T65879 CWS37O 42618140 IC50 = 7943.28 nM T65879 CQE43D 42618141 IC50 = 3981.07 nM T65879 C2IK0N 42618142 IC50 = 12589.25 nM T65879 C2JV3O 42618143 IC50 = 6309.57 nM T65879 CG01BO 42618144 IC50 = 2511.89 nM T65879 CCSQ57 42618145 IC50 = 10000 nM T65879 CW7X6L 42618146 IC50 > 25118.86 nM T65879 C4K6PD 42618147 IC50 > 25118.86 nM T65879 C5SL3N 42618148 IC50 = 15848.93 nM T65879 CYU47O 42618149 IC50 > 25118.86 nM T65879 CWD4R1 42618150 IC50 = 12589.25 nM T65879 C5X2UV 42618151 IC50 = 25118.86 nM T65879 CIN5U6 42618152 IC50 > 25118.86 nM T65879 CW8VP1 42618153 IC50 = 3981.07 nM T65879 CCB0L2 42618154 IC50 = 3162.28 nM T65879 CC7GS2 42618155 IC50 = 12589.25 nM T65879 CZ86OF 42618156 IC50 = 5011.87 nM T65879 CX9N3L 42618157 IC50 = 10000 nM T65879 C38FZM 42618158 IC50 = 15848.93 nM T65879 C2I7HC 42618159 IC50 = 10000 nM T65879 C6YSW0 42618160 IC50 = 19952.62 nM T65879 C3IY4O 42618161 IC50 > 25118.86 nM T65879 C1CY8R 42618162 IC50 > 25118.86 nM T65879 C80KDA 42618163 IC50 > 25118.86 nM T65879 CG28AW 42618164 IC50 > 25118.86 nM T65879 CO4FV0 42630578 IC50 = 3162.28 nM T65879 C90BUF 43157763 IC50 > 100000 nM T65879 CJ7D5T 43157843 IC50 > 100000 nM T65879 C6Z2SA 43560957 IC50 > 100000 nM T65879 CO42DC 44138048 IC50 > 10000 nM T65879 CL65QV 44138049 IC50 > 10000 nM T65879 CLW80F 44160269 IC50 = 35000 nM T65879 C6RN7P 44187181 IC50 = 7 nM T65879 CI4Y7O 44187182 IC50 = 7 nM T65879 C6LTC3 44187183 IC50 = 12 nM T65879 CK73NR 44219749 IC50 > 50000 nM T65879 CBE4N3 44317538 IC50 > 20000 nM T65879 CC9FJ1 44317726 IC50 > 20000 nM T65879 CGU68A 44317768 IC50 > 20000 nM T65879 CO4AW6 44317844 IC50 > 20000 nM T65879 CBR5L9 44317865 IC50 > 20000 nM T65879 CKJ9W8 44317866 IC50 > 20000 nM T65879 CMI34Q 44353870 IC50 = 1698 nM T65879 CSEY31 44353885 IC50 = 1479 nM T65879 CR13ES 44353890 IC50 = 3981 nM T65879 CI3U0J 44353891 IC50 = 2692 nM T65879 CA16WX 44353923 IC50 = 3090 nM T65879 CIJ19R 44353953 IC50 = 3981 nM T65879 CCLG72 44353954 IC50 = 1096 nM T65879 CO97FH 44353955 IC50 = 851 nM T65879 C86QXB 44353966 IC50 = 1230 nM T65879 C15JMN 44353967 IC50 = 2089 nM T65879 CLV7G6 44353968 IC50 = 1622 nM T65879 C8RZV9 44353969 IC50 = 2344 nM T65879 CN91IA 44353987 IC50 = 155 nM T65879 CGB6I4 44353995 IC50 = 245 nM T65879 CJIC08 44353996 IC50 = 1202 nM T65879 C7MS0Y 44353999 IC50 = 5129 nM T65879 CW5J2M 44354000 IC50 = 1175 nM T65879 CY6K7E 44354001 IC50 = 2344 nM T65879 CFO54D 44354009 IC50 = 4074 nM T65879 C7HBR2 44354029 IC50 = 331 nM T65879 CJD42L 44354030 IC50 = 3802 nM T65879 CS7N9Y 44406379 IC50 = 1200 nM T65879 CAW8D0 44406386 IC50 = 1200 nM T65879 C9LVS2 44406419 IC50 = 150 nM T65879 CRC9U2 44406468 IC50 = 3800 nM T65879 COQ56E 44406470 IC50 = 3700 nM T65879 C4HSU0 44406486 IC50 = 5000 nM T65879 C47WRS 44406506 IC50 > 100000 nM T65879 CS60YA 44406549 IC50 = 500 nM T65879 C1GJF8 44406564 IC50 = 400 nM T65879 CG5T2C 44406565 IC50 = 30 nM T65879 CM58DH 44406581 IC50 = 30000 nM T65879 CG3CW4 44406586 IC50 = 30 nM T65879 CPR69I 44406614 IC50 = 700 nM T65879 C1IT5S 44406634 IC50 = 100 nM T65879 C51NLK 44406635 IC50 = 500 nM T65879 CMX18H 44406636 IC50 = 1000 nM T65879 CL7M1J 44425584 IC50 = 1995.26 nM T65879 C2C5OI 44425585 IC50 = 1000 nM T65879 CZ67YJ 44425588 IC50 = 1000 nM T65879 C9KTQ7 44425594 IC50 = 630.96 nM T65879 CXV8D5 44425596 IC50 = 794.33 nM T65879 CI26BP 44425599 IC50 = 1000 nM T65879 C1GY8L 44425606 IC50 = 794.33 nM T65879 CMN54H 44442024 IC50 = 3860 nM T65879 CX4M1T 44448398 IC50 = 6700 nM T65879 C0HML9 44448550 IC50 = 2990 nM T65879 C0VS4B 44448553 IC50 = 4840 nM T65879 CL2U8A 44448587 IC50 = 1910 nM T65879 C1I5OF 44448662 IC50 = 731 nM T65879 C01RDH 44448700 IC50 = 146 nM T65879 C9IGA2 44449047 IC50 = 2630 nM T65879 CN0K9Q 44449188 IC50 = 850 nM T65879 C4WRN5 44541014 IC50 = 50 nM T65879 CA78EV 44573281 IC50 = 9700 nM T65879 CCL85F 44575073 IC50 > 50000 nM T65879 CJX06P 44575126 IC50 > 50000 nM T65879 CE8FC7 44575127 IC50 > 50000 nM T65879 C3B9XA 44591531 IC50 = 316.23 nM T65879 CVI6S3 44591532 IC50 = 31.62 nM T65879 C06RIF 44591552 IC50 = 794.33 nM T65879 CCD3F9 44591553 IC50 = 1258.93 nM T65879 CXP21B 44591574 IC50 = 125.89 nM T65879 C4T8XR 44591575 IC50 = 12.59 nM T65879 CHQR35 44591576 IC50 = 1000 nM T65879 C28QLM 44605035 IC50 > 50000 nM T65879 C75XHS 44605037 IC50 > 50000 nM T65879 CU3RF1 45139989 IC50 > 10000 nM T65879 CQGZ06 45139991 IC50 > 10000 nM T65879 CW4LQ3 45267192 IC50 = 25 nM T65879 C29EIZ 45268050 IC50 = 39 nM T65879 CAXI74 45268940 IC50 = 22 nM T65879 CST87Y 45269780 IC50 = 14 nM T65879 C2JVA4 45270368 IC50 = 32 nM T65879 CCNU16 45270611 IC50 = 11 nM T65879 C76TRL 45270614 IC50 = 79 nM T65879 CL45SW 45271427 IC50 = 43 nM T65879 C1SAJ4 45272329 IC50 = 8 nM T65879 CX0A2G 45273193 IC50 = 44 nM T65879 CZ58FY 46215814 IC50 = 100 nM T65879 CY3HW5 46224684 IC50 = 33 nM T65879 C7ON5A 46233287 IC50 > 10000 nM T65879 CJOM49 46880136 IC50 > 50000 nM T65879 CQR9K1 46933384 IC50 = 40000 nM T65879 C83VHI 49864785 IC50 = 4600 nM T65879 C2UTK6 49864850 IC50 = 2200 nM T65879 CAE53W 49865153 IC50 > 4000 nM T65879 CF5B1D 49865328 IC50 > 100000 nM T65879 CG4TE7 49865330 IC50 > 100000 nM T65879 CH2I3A 50941935 IC50 = 420 nM T65879 CIB60D 50941936 IC50 = 230 nM T65879 CP91XJ 51346795 IC50 > 100000 nM T65879 CEQN27 52936621 Ki > 1000 nM T65879 C5QCR2 53317336 IC50 = 9000 nM T65879 CV1T5R 53321248 IC50 > 100000 nM T65879 C1O4MK 53321249 IC50 > 100000 nM T65879 C6IS2B 53323910 IC50 = 41000 nM T65879 CUG3D4 53325187 IC50 > 100000 nM T65879 C8ZRE3 53356518 IC50 > 50000 nM T65879 CIK9F2 54580282 IC50 = 15848.93 nM T65879 C8R0GT 54581284 IC50 = 5011.87 nM T65879 C5V6OY 54582175 IC50 > 30000 nM T65879 CF5TS9 54585210 IC50 > 15848.93 nM T65879 CNUP53 54586040 IC50 = 20370 nM T65879 CE2XK3 54587170 IC50 = 12589.25 nM T65879 C9EMO2 54765177 IC50 = 330 nM T65879 C1WJD3 59406184 IC50 = 79.43 nM T65879 CS8F3Q 59406262 IC50 = 158.49 nM T65879 CVY3C8 59406271 IC50 = 7.943 nM T65879 CSPD01 59744353 IC50 = 251.19 nM T65879 CC8T7R 59744382 IC50 = 316.23 nM T65879 CM1S2I 59744412 IC50 = 316.23 nM T65879 C0SBK4 59744417 IC50 = 25.12 nM T65879 C6PB3C 59744422 IC50 = 6.31 nM T65879 C7JDY6 59744451 IC50 = 6.31 nM T65879 C8Q2MN 59744508 IC50 = 6.31 nM T65879 C56DCI 59744533 IC50 = 100 nM T65879 CMB8X7 59744546 IC50 = 199.53 nM T65879 C23NOS 59744560 IC50 = 398.11 nM T65879 C4QLN7 59744593 IC50 = 50.12 nM T65879 C1MR8Q 60097495 IC50 > 10000 nM T65879 CL36SQ 61992242 IC50 > 100000 nM T65879 CNP85L 61992815 IC50 > 100000 nM T65879 CU28AB 62900145 IC50 > 100000 nM T65879 CV63UL 67240318 IC50 > 10000 nM T65879 CQ8HE2 70690944 IC50 > 30000 nM T65879 C13FWG 70695135 IC50 > 30000 nM T65879 C0VZB2 70697173 IC50 > 30000 nM T65879 CQ31PG 71138120 Ki > 30000 nM T65879 CA2V1U 71462267 IC50 = 31.62 nM T65879 CB04OD 82482456 IC50 > 100000 nM T65879 C75AVW 102334651 Ki = 800 nM T65879 CQCX41 118737057 IC50 = 353 nM T65879 C0EJS9 129320519 Ki = 650 nM T65879 C2AN7T 134611886 IC50 > 100000 nM T65879 C54FXD 134957362 IC50 > 10000 nM T65879 CKHV90 135401952 IC50 = 5011.87 nM T65879 CD8V9X 135432858 IC50 = 25 nM T65879 CRY3K8 135456003 IC50 = 20000 nM T65879 C86WCU 135469510 IC50 > 20000 nM T65879 CV76UY 135909516 IC50 = 15848.93 nM T65879 CR83YE 137631544 Ki = 2000 nM T65879 CT0P5R 137632102 Ki = 16000 nM T65879 C5CU9T 137632103 Ki > 30000 nM T65879 C6FJ1P 137632317 Ki = 5300 nM T65879 CB9XT2 137632532 Ki = 1500 nM T65879 C6W2PJ 137633160 Ki = 1400 nM T65879 CDBV08 137634477 Ki = 2000 nM T65879 C0KU4C 137635130 Ki = 1600 nM T65879 C8F7OK 137636751 Ki > 30000 nM T65879 CVZ5Y6 137637765 Ki = 2400 nM T65879 CK08TL 137640054 Ki = 5300 nM T65879 C3FNV9 137640501 Ki = 13000 nM T65879 C8BF9I 137640852 Ki > 30000 nM T65879 C02MPZ 137641352 Ki = 1700 nM T65879 C2L6ZU 137641677 Ki = 80 nM T65879 C1Y6NI 137641784 Ki = 2500 nM T65879 C7BQX5 137642493 Ki = 15000 nM T65879 CSZ6B9 137643197 Ki > 30000 nM T65879 CC0T7J 137644890 Ki = 2100 nM T65879 C2QSP4 137645617 Ki = 1800 nM T65879 CS9T4Q 137646916 Ki = 3100 nM T65879 C5P2NR 137648275 Ki > 30000 nM T65879 CA84NC 137648771 Ki = 10000 nM T65879 CH2S7I 137648911 Ki > 30000 nM T65879 C5QMA7 137648912 Ki > 30000 nM T65879 C2AN5P 137650396 Ki = 5300 nM T65879 CKW51R 137650911 Ki > 30000 nM T65879 C6VHT8 137651289 Ki > 30000 nM T65879 CS9WT0 137651927 Ki = 13000 nM T65879 C6L5KV 137652726 Ki > 30000 nM T65879 CZ1L7Y 137653022 Ki = 2400 nM T65879 C1G3KP 137653092 Ki > 30000 nM T65879 CP5X0N 137653110 Ki = 5300 nM T65879 C5TJ8K 137653144 Ki = 9800 nM T65879 C9AIU6 137655282 Ki = 2900 nM T65879 C0M4KH 137655668 Ki > 30000 nM T65879 CGKU15 137655801 Ki > 30000 nM T65879 CE8N2X 137655941 Ki = 1000 nM T65879 CYKL36 137656635 Ki > 30000 nM T65879 CF41YQ 137656752 Ki = 7700 nM T65879 C86SIX 137657214 Ki = 1700 nM T65879 C3VT5X 137657569 Ki > 30000 nM T65879 CA7RD3 137657800 Ki = 1600 nM T65879 C7S2EH 137657801 Ki = 6000 nM T65879 COXH36 137659346 Ki = 16000 nM T65879 C2BRJ0 137659655 Ki = 16000 nM T65879 CCNA02 137660360 Ki > 30000 nM T65879 COS48M 137661213 Ki > 30000 nM T65879 C9O3EJ 137661645 Ki = 10000 nM T65879 CLBV34 137661772 Ki = 12100 nM T65879 CT89FP 145952913 IC50 = 35500 nM T65879 CW3RV1 145953992 IC50 = 2511.89 nM T65879 CCL34O 145954234 IC50 = 125.89 nM T65879 C4ZH8E 145954241 IC50 = 158.49 nM T65879 CNT8O5 145954713 IC50 = 199.53 nM T65879 CB0F7N 145955167 IC50 = 158.49 nM T65879 CJDG56 145960632 IC50 > 31622.78 nM T65879 CB7TW3 145960672 IC50 = 158.49 nM T65879 CH6G1S 145960935 IC50 = 100 nM T65879 C6ZJQ4 145961055 IC50 = 125.89 nM T65879 CE21QP 145961382 IC50 > 25118.86 nM T65879 CQ9FN7 145961544 IC50 = 2511.89 nM T65879 C23GXR 145961663 IC50 = 79.43 nM T65879 CJ0K8Z 145962062 IC50 = 125.89 nM T65879 CV0T1U 145962184 IC50 = 31.62 nM T65879 CA2RO4 145962531 IC50 = 2511.89 nM T65879 CCL79I 145963000 IC50 = 79.43 nM T65879 CI0V8W 145963248 IC50 > 25118.86 nM T65879 C0JX1P 145963398 IC50 = 3162.28 nM T65879 CJZ4G3 145963549 IC50 = 79.43 nM T65879 C9V6AQ 145963687 IC50 = 158.49 nM T65879 C91BHP 145971744 IC50 > 100000 nM T65879 CML8O0 145979124 IC50 > 100000 nM T65879 CQLH68 145979774 IC50 > 100000 nM T65879 C5YR8W 145979893 IC50 > 100000 nM T65879 CGL48D 145980076 IC50 > 100000 nM T65879 C5LK9A 145980083 IC50 > 100000 nM T65879 CCSY15 145980681 IC50 > 100000 nM T65879 CY80PH 145981483 IC50 > 100000 nM T65879 CN3U5W 145981500 IC50 > 100000 nM T65879 CFSQ94 145981688 IC50 > 100000 nM T65879 CI3P2B 145981824 IC50 > 100000 nM T65879 CVRZ23 145984375 IC50 > 100000 nM T65879 CGE7B8 145987124 IC50 > 100000 nM T65879 C86HGI 145987159 IC50 > 100000 nM T65879 CU3J8R 145987461 IC50 > 100000 nM T65879 CRJQ18 145988918 IC50 > 100000 nM T65879 C8QH2W 145989390 IC50 > 100000 nM T65879 CFAK86 145989643 IC50 > 100000 nM T65879 CHWR01 145989760 IC50 > 100000 nM T65879 C3EIA1 145990026 IC50 > 100000 nM T65879 CBZ94U 145990465 IC50 > 100000 nM T65879 C8M5AU 145990524 IC50 = 34900 nM T65879 C4FQ0C 145990918 IC50 > 100000 nM T65879 CN38UG 145990988 IC50 > 100000 nM T65879 CGSZ75 145991182 IC50 > 100000 nM T65879 C2SY4M 145991367 IC50 > 100000 nM T65879 C0CJ9I 145991401 IC50 > 100000 nM T65879 CI60XK 145991710 IC50 > 100000 nM T65879 C17TOS 145991715 IC50 > 100000 nM T65879 C68ZYI 145991820 IC50 > 100000 nM T65879 C3HIB8 145992014 IC50 > 100000 nM T65879 CF28WP 145992122 IC50 > 100000 nM T65879 C85OWM 145992355 IC50 > 100000 nM T65879 CD54KY 145992596 IC50 > 100000 nM T65879 CQI81V 145992947 IC50 > 100000 nM T65879 C3NU7C 145993088 IC50 > 100000 nM T65879 C0CJ9B 145993626 IC50 > 100000 nM T65879 C2GH5C 145993662 IC50 > 100000 nM T65879 CMJ6G4 145993951 IC50 > 100000 nM T65879 C2MD1Q 155513187 IC50 > 10000 nM T65879 C2CG1A 155537016 IC50 > 10000 nM T65879 D00ERW 44444843 Ki > 3750 nM T65879 D00HVA 11624601 Ki > 1500 nM T65879 D00XDG 11708263 IC50 > 30000 nM T65879 D00YTQ 9926054 IC50 = 4000 nM T65879 D01OBJ 11414735 IC50 = 1000 nM T65879 D01YWE 25207521 IC50 > 50000 nM T65879 D03OKV 9844320 IC50 > 10000 nM T65879 D06WGX 9549184 IC50 > 25000 nM T65879 D07ADX 54764565 IC50 = 591 nM T65879 D07MQC 9949093 IC50 = 100 nM T65879 D0EU1R 46215815 IC50 > 25118 nM T65879 D0F0VD 135465539 IC50 = 250 nM T65879 D0F8QJ 5281813 IC50 > 10000 nM T65879 D0LE7J 58221375 IC50 > 100000 nM T65879 D0Q3NG 11715520 Ki > 1500 nM T65879 D0R6FJ 64961 IC50 = 15000 nM T65879 D0S7IE 11658882 Ki = 970 nM T65879 D0UP6G 11600944 IC50 > 15848.93 nM T85421 D04AHQ 71721540 IC50 = 470 nM T85421 D0M0XB 10302451 IC50 > 10000 nM T85421 D0X4MN 11597537 IC50 = 200 nM T85421 D0WS1V 448991 IC50 > 10000 nM T85421 D09QKG 25104303 IC50 = 3000 nM T85421 D0PO8N 117881270 IC50 = 1300 nM T85421 CWZ2V1 619002 IC50 = 2300 nM T85421 CVN83J 656950 IC50 > 10000 nM T85421 C72CNT 2747117 EC50 = 12400 nM T85421 C2TAD3 3036289 EC50 = 1240 nM T85421 CL5I2U 5330279 IC50 > 10000 nM T85421 CA32PV 6540289 IC50 > 30000 nM T85421 C38UZJ 6852206 EC50 = 890 nM T85421 C3JEN8 9543521 IC50 = 2500 nM T85421 C2OL7K 9796455 IC50 > 50000 nM T85421 CM5Z8X 9869943 IC50 > 1000 nM T85421 CN0AJ9 9934347 EC50 = 41 nM T85421 CJO47T 9948405 IC50 > 10000 nM T85421 C2W3AV 9995236 IC50 = 1000 nM T85421 CV8I5X 9999342 IC50 > 10000 nM T85421 C5TQ7X 10247543 IC50 > 10000 nM T85421 C8RD3V 10301884 IC50 > 10000 nM T85421 C2WQ8M 10473563 IC50 > 10000 nM T85421 C43NPS 11373886 IC50 > 10000 nM T85421 C0H6QS 11495680 IC50 > 10000 nM T85421 CIW9L5 11502867 IC50 > 10000 nM T85421 C7H6PZ 11516913 EC50 = 910 nM T85421 CK2Q0X 11516978 IC50 > 10000 nM T85421 CPE53F 11526238 IC50 > 10000 nM T85421 C5BM4T 11531799 IC50 > 10000 nM T85421 C53OSD 11532048 IC50 > 10000 nM T85421 CC4QM5 11532676 IC50 > 10000 nM T85421 CTG83F 11539329 Ki = 9 nM T85421 C01FVM 11546457 IC50 > 10000 nM T85421 CM57ZU 11553156 EC50 > 10000 nM T85421 C4I0YH 11558900 EC50 = 2500 nM T85421 C3KT8X 11559766 EC50 = 1600 nM T85421 CNBM81 11562171 IC50 > 10000 nM T85421 C6O0HX 11587896 EC50 = 1400 nM T85421 C24JGU 11589125 EC50 = 1400 nM T85421 CQ82SM 11589163 EC50 = 3900 nM T85421 CMIL86 11590363 Ki = 13 nM T85421 C0NV9Y 11596881 IC50 > 10000 nM T85421 CUK87R 11602023 EC50 = 3400 nM T85421 CQ29WV 11602291 EC50 = 1400 nM T85421 C1BLZ5 11620055 IC50 > 10000 nM T85421 C9NP0W 11638309 IC50 = 850 nM T85421 C9T6SC 11640926 Ki = 4 nM T85421 C6NO5B 11647280 EC50 = 280 nM T85421 C24GRQ 11661959 IC50 > 10000 nM T85421 CS72ED 11682843 IC50 > 10000 nM T85421 CLC53E 11691173 IC50 > 10000 nM T85421 C2CPZ3 11695458 EC50 = 5500 nM T85421 C1FTX3 11719305 IC50 > 10000 nM T85421 CFHX82 11837140 IC50 = 700 nM T85421 CBC08P 11846124 IC50 = 530 nM T85421 CD60CH 11846125 IC50 = 110 nM T85421 C5LIW2 11846126 IC50 = 1200 nM T85421 CNJB87 11846287 IC50 > 10000 nM T85421 CEMS06 11846288 IC50 > 10000 nM T85421 C7DI3U 11846294 IC50 = 5800 nM T85421 CIJ93W 11846459 IC50 = 640 nM T85421 C5KC7Q 11846461 IC50 = 1100 nM T85421 CFPW41 16007116 IC50 = 480 nM T85421 C3V6EX 16049812 IC50 = 250 nM T85421 C6L9VD 16216351 IC50 = 560 nM T85421 CM2UY0 23647201 IC50 = 16400 nM T85421 C3UOY0 23647202 IC50 > 30000 nM T85421 CGRL48 23647204 IC50 > 30000 nM T85421 CF3XS2 23647210 IC50 = 19400 nM T85421 C7HF9E 23647211 IC50 = 10600 nM T85421 CQ87FP 23647212 IC50 = 5600 nM T85421 CNOA35 23647216 IC50 = 32000 nM T85421 CQDB80 23647217 IC50 = 26600 nM T85421 C1MYT5 23647218 IC50 > 30000 nM T85421 CS69RG 23647219 IC50 > 30000 nM T85421 CKP16G 23647223 IC50 = 14700 nM T85421 C0PXL4 23647225 IC50 > 30000 nM T85421 C5AHM8 23647226 IC50 > 30000 nM T85421 C0E4ZY 23647227 IC50 > 30000 nM T85421 CY3L0H 23647228 IC50 > 30000 nM T85421 CM10AZ 23647229 IC50 > 30000 nM T85421 C29TJW 23647230 IC50 > 30000 nM T85421 C4NL5H 23647231 IC50 > 30000 nM T85421 C62DWL 23647232 IC50 > 30000 nM T85421 C7C4IX 23647233 IC50 > 30000 nM T85421 C4W5GQ 23647234 IC50 > 30000 nM T85421 C8QE9S 23647235 IC50 > 30000 nM T85421 CR2V5H 23647236 IC50 > 30000 nM T85421 CGXB32 23647237 IC50 = 410 nM T85421 CG6D4M 23647319 IC50 > 10000 nM T85421 CY8Z7X 23647330 IC50 > 10000 nM T85421 C4XD8H 23647348 IC50 > 10000 nM T85421 CJ7M8K 24823663 IC50 = 1300 nM T85421 CLP68C 24823665 IC50 = 790 nM T85421 CRV5C7 24823814 IC50 = 1500 nM T85421 CSW3D9 24823964 IC50 = 1800 nM T85421 CL61YV 24824104 IC50 = 540 nM T85421 C42HGN 24957306 IC50 = 2700 nM T85421 CK4W5P 24957308 IC50 = 2000 nM T85421 CE8KJ9 24960632 IC50 = 8200 nM T85421 C9WOQ0 24960635 IC50 = 2300 nM T85421 C6B0IM 24961360 IC50 = 3100 nM T85421 CM2K9V 25119432 IC50 = 4300 nM T85421 CYTV68 25181985 IC50 = 560 nM T85421 C5KIE7 25182113 IC50 = 1000 nM T85421 C0E5HT 44313624 IC50 = 3200 nM T85421 CV09DY 44410717 IC50 > 10000 nM T85421 CP3CI1 44410720 IC50 > 10000 nM T85421 C8W7AD 44410723 IC50 > 10000 nM T85421 CAT5X4 44410829 IC50 > 10000 nM T85421 CC6Y5P 44410844 IC50 > 10000 nM T85421 CG34TY 44410851 IC50 > 10000 nM T85421 C41EIA 44410869 IC50 > 10000 nM T85421 CB6AE8 44410948 IC50 > 10000 nM T85421 CXZG12 44410949 IC50 > 10000 nM T85421 CS7IE9 44410953 IC50 > 10000 nM T85421 CA9M4X 44410954 IC50 > 10000 nM T85421 C3SP5H 44410955 IC50 > 10000 nM T85421 C5D6YP 44410956 IC50 > 10000 nM T85421 C5W1VC 44410959 IC50 > 10000 nM T85421 CM1C2G 44410960 IC50 > 10000 nM T85421 CVSI80 44411048 IC50 > 10000 nM T85421 CN72BR 44411161 IC50 > 10000 nM T85421 C4AW0O 44411183 IC50 > 10000 nM T85421 CY6EW5 44419110 IC50 = 1890 nM T85421 CP05HO 44419116 IC50 = 5700 nM T85421 C9IWT5 44419118 IC50 = 7360 nM T85421 CNJ5F1 44419119 IC50 = 5240 nM T85421 CAYL35 44419128 IC50 = 1200 nM T85421 COC4P2 44419129 IC50 = 2700 nM T85421 C5ZMS7 44419130 IC50 > 10000 nM T85421 CH8WZ7 44419135 IC50 = 9400 nM T85421 CRI6V9 44419136 IC50 = 1800 nM T85421 CY6DK0 44419137 IC50 > 10000 nM T85421 CZP46I 44419138 IC50 > 10000 nM T85421 CQT30U 44419143 IC50 = 10500 nM T85421 C8J6MZ 44419144 IC50 = 610 nM T85421 CYM3X7 44419145 IC50 = 8300 nM T85421 CHG96R 44419146 IC50 > 10000 nM T85421 CLX1B5 44419150 IC50 = 4300 nM T85421 C0CLT1 44419151 IC50 > 10000 nM T85421 CKL2A8 44419152 IC50 = 5900 nM T85421 CJ1RE0 44419155 IC50 = 10800 nM T85421 C65XAW 44419156 IC50 = 8010 nM T85421 CMCF90 44419158 IC50 = 2600 nM T85421 C40QDE 44419161 IC50 = 7300 nM T85421 CNX3P1 44419163 IC50 > 10000 nM T85421 C1XI7E 44419168 IC50 > 10000 nM T85421 CDIL57 44419169 IC50 = 890 nM T85421 C4YQD8 44419170 IC50 > 10000 nM T85421 CQE6D3 44419174 IC50 = 5500 nM T85421 C76JCA 44419175 IC50 = 350 nM T85421 CK4Z6B 44419182 IC50 = 5300 nM T85421 CST57V 44419183 IC50 > 2500 nM T85421 C1RL3U 44419191 IC50 = 2900 nM T85421 C8IJ2U 44419202 IC50 = 700 nM T85421 C5KBX0 44419203 IC50 = 490 nM T85421 CP1C8D 44419211 IC50 = 490 nM T85421 CO9AK1 44419214 IC50 = 4630 nM T85421 CE20PN 44419215 IC50 = 6920 nM T85421 C4V6YN 44419216 IC50 = 1200 nM T85421 CF4I1R 44419217 IC50 = 620 nM T85421 C13EQD 44419220 IC50 > 10000 nM T85421 C1KQL5 44419221 IC50 = 807 nM T85421 CD8EB4 44419222 IC50 = 480 nM T85421 CY1Q7N 44419226 IC50 = 1400 nM T85421 CXR83C 44419227 IC50 = 7540 nM T85421 CMKH90 44591675 IC50 = 920 nM T85421 C2X7DJ 44591676 IC50 = 840 nM T85421 CUL5A2 44591677 IC50 = 1100 nM T85421 C2S4PZ 44591703 IC50 = 460 nM T85421 COZ16T 44591706 IC50 = 3500 nM T85421 CHD64X 44591707 IC50 = 357 nM T85421 C8T1LV 44591735 IC50 = 814 nM T85421 CV26OD 44591737 IC50 = 221 nM T85421 CY26UI 44591738 IC50 = 6020 nM T85421 C3D8RZ 44591739 IC50 = 245 nM T85421 C5Z3LI 44591740 IC50 = 98 nM T85421 C6OZB5 44591767 IC50 = 209 nM T85421 CU23PY 44591768 IC50 = 114 nM T85421 COHK45 44591769 IC50 = 299 nM T85421 C1LD0P 50943125 IC50 = 220 nM T85421 CI0Z7D 50943202 IC50 = 1700 nM T85421 CHIY40 50943203 IC50 = 290 nM T85421 CGZC83 50943588 IC50 = 710 nM T85421 CEX3H8 50943666 IC50 = 200 nM T85421 C1JY2U 50943668 IC50 = 820 nM T85421 CPS4I5 50943669 IC50 = 240 nM T85421 C83EZX 50943670 IC50 = 700 nM T85421 CNUZ80 50943753 IC50 = 1300 nM T85421 COU4W2 50943754 IC50 = 650 nM T85421 C2J7ZP 50943755 IC50 = 1300 nM T85421 CTO6N5 56834943 IC50 = 350 nM T85421 CHU75J 57390951 IC50 = 2500 nM T85421 CG51FX 57392289 IC50 = 300 nM T85421 CSYJ61 57392738 IC50 = 500 nM T85421 C2IZ3W 57392739 IC50 = 91 nM T85421 C9P1SC 57393560 IC50 = 240 nM T85421 C03CNR 57394466 IC50 = 440 nM T85421 CX9B4S 57394467 IC50 = 1800 nM T85421 C1EYU6 57394468 IC50 = 1200 nM T85421 CW7XA9 57397040 IC50 = 210 nM T85421 C4V9RN 57398023 IC50 = 200 nM T85421 CZI7A2 57398024 IC50 = 230 nM T85421 C4RJ0E 57398025 IC50 = 1600 nM T85421 CE76QR 57399681 IC50 = 200 nM T85421 CLI72R 57401441 IC50 = 860 nM T85421 CPY13U 57401443 IC50 = 1700 nM T85421 CKE0V9 57403185 IC50 = 1700 nM T85421 CY8HG6 58017084 IC50 = 1100 nM T85421 C5IN0E 59718933 IC50 = 4900 nM T85421 C1XCV6 59718972 IC50 = 3300 nM T85421 C20CME 59743327 IC50 = 1000 nM T85421 C4IM1V 59743368 IC50 = 1400 nM T85421 C6VYE9 59743400 IC50 = 980 nM T85421 CJE42G 59743404 IC50 = 12000 nM T85421 CUW7J8 59743407 IC50 = 240 nM T85421 C8L4KY 59743442 IC50 = 960 nM T85421 CSK8O7 59743445 IC50 = 580 nM T85421 C0MO4E 59743458 IC50 > 30000 nM T85421 C5UYK1 59743461 IC50 = 590 nM T85421 CWB21E 59743477 IC50 = 1100 nM T85421 C5RH4P 59743505 IC50 = 1400 nM T85421 C3KY7N 59743507 IC50 = 1100 nM T85421 CJ2NM1 59743549 IC50 = 2000 nM T85421 CY89OP 59743571 IC50 = 350 nM T85421 CDA46Z 59846170 IC50 = 830 nM T85421 C86QAW 59846186 IC50 = 2500 nM T85421 C20GMT 59846188 IC50 = 1700 nM T85421 C24GXO 59846214 IC50 = 2700 nM T85421 CO8R0G 59846284 IC50 = 860 nM T85421 CVZ67M 66816803 IC50 = 4200 nM T85421 CLG56W 66940332 IC50 = 420 nM T85421 CF7N8W 71454040 IC50 = 4700 nM T85421 CU0EG4 71457558 IC50 = 430 nM T85421 CAK95D 71461189 IC50 = 4300 nM T85421 CTL1H9 71655707 IC50 = 104 nM T85421 CH4DI3 90667139 EC50 = 23 nM T85421 CQ2G3S 91754590 IC50 < 50 nM T85421 CY82JT 118146747 IC50 = 1015 nM T85421 CET9N4 118146870 IC50 < 50 nM T85421 C4PBE7 118146871 IC50 = 990 nM T85421 C4Q5CE 135453643 Ki < 1000000 nM T85421 C1EU9T 155514086 IC50 = 500 nM T85421 CGD3P5 155521400 IC50 = 600 nM T85421 C97IKV 155525801 IC50 = 3300 nM T85421 C93WEV 155536948 IC50 = 2700 nM T85421 CM8N5C 155538719 IC50 = 6700 nM T85421 C8SA9Q 155539342 IC50 = 2100 nM T85421 C0ESP6 155542557 IC50 = 900 nM T85421 CEK8L7 155548073 IC50 = 4500 nM T85421 C6EXG0 155555966 IC50 = 11100 nM T85421 CC47QL 155561957 IC50 = 2500 nM T85421 C6H4AW 155565897 IC50 = 1200 nM T85421 CM92KO 155569233 IC50 = 4300 nM T85421 D00HVA 11624601 Ki = 4 nM T85421 D02PVB 8515 IC50 = 3400 nM T85421 D02XHC 448912 IC50 = 3300 nM T85421 D05QJS 5480230 EC50 = 158 nM T85421 D07IHM 9823787 IC50 > 30000 nM T85421 D07OAT 456214 IC50 > 1000 nM T85421 D09QBA 23378546 IC50 > 30000 nM T85421 D0H0OO 25075991 EC50 = 87 nM T85421 D0Q3NG 11715520 Ki = 440 nM T85421 D0S7IE 11658882 Ki = 1900 nM T85421 D0UG5M 9956146 EC50 = 5 nM T70508 C97TNH 10177 IC50 = 2200 nM T70508 D07IHM 9823787 IC50 > 10000 nM T70508 D09QBA 23378546 IC50 > 10000 nM T59537 D0E6XR 3062316 Ki = 0.5 nM T59537 D0OB0F 5328940 Ki = 12.7 nM T59537 D02KKA 24856436 Ki = 470 nM T59537 D0M0XB 10302451 Ki = 39.8 nM T59537 D0H8KG 5311382 Ki = 0.8 nM T59537 CP71KC 683649 IC50 = 1200 nM T59537 CTQ48P 9927432 Ki = 16.85 nM T59537 CJ9KN7 11683817 IC50 > 10000 nM T59537 C6EU9X 16048415 Ki = 5520 nM T59537 C6ZVL0 24856612 Ki = 470 nM T59537 C63ILA 24896610 Ki = 48.47 nM T59537 CGW79M 42609478 Ki = 0.5 nM T59537 CO8X1V 44418540 Ki = 521.5 nM T59537 CNK03V 44526249 Ki = 10.94 nM T59537 C7TO2X 44526759 Ki = 32.4 nM T59537 C3DJQ4 44526801 Ki = 25.68 nM T59537 CVF38O 44529068 Ki = 720.2 nM T59537 CREB48 44532315 Ki = 67.19 nM T59537 C3VRO9 44557921 IC50 > 10000 nM T59537 C4UPO3 57400258 EC50 = 18 nM T59537 CQU6T8 145983754 Ki = 32.4 nM T59537 CL0WX3 145986228 Ki = 51.73 nM T59537 CQ57PG 155513251 Ki = 39.8 nM T59537 CROW39 155518316 IC50 = 9332.54 nM T59537 CLV43W 155520629 Ki = 48.47 nM T59537 C5RHO2 155523681 IC50 = 1548.82 nM T59537 C8Y3IK 155527161 IC50 = 6309.57 nM T59537 C3DW7P 155559865 IC50 = 616.6 nM T59537 D03NPX 447077 Ki = 43.65 nM T59537 D0D5EW 5311104 Ki = 10.4 nM T59537 D0S1KJ 5328733 Ki = 2.3 nM T59537 D0ZH1U 2051 Ki = 1870 nM T87670 D0O1UZ 644019 EC50 = 445 nM T87670 D0O3OS 104850 EC50 = 2010 nM T87670 D0P1FO 16078 EC50 = 14200 nM T87670 C0ZR5B 4407 EC50 > 20000 nM T87670 CVL1A0 320263 IC50 > 10000 nM T87670 CL3UD5 320264 IC50 > 10000 nM T87670 CFY02L 356017 IC50 > 10000 nM T87670 C8X7ST 356018 IC50 > 10000 nM T87670 C3Q4CT 375895 EC50 > 20000 nM T87670 CJ37RB 378629 EC50 = 2700 nM T87670 CGT6F3 738959 IC50 > 10000 nM T87670 C0MYU2 1281700 IC50 > 10000 nM T87670 C8KD9F 1281702 IC50 = 5090 nM T87670 CH8PY0 1281704 IC50 > 10000 nM T87670 CX5F6G 1281706 IC50 > 10000 nM T87670 C63LER 2958539 EC50 = 55.7 nM T87670 CVA6B4 2964166 EC50 = 218 nM T87670 CX7RC9 4929019 EC50 = 5.6 nM T87670 CR0A8U 4930011 EC50 = 19.4 nM T87670 CJTG76 4932893 EC50 = 175.7 nM T87670 C7WJE8 5177252 EC50 = 6.2 nM T87670 CR03OP 5185091 EC50 = 39.2 nM T87670 CC4B0K 5917569 IC50 > 10000 nM T87670 CE6M2A 6294602 EC50 = 600 nM T87670 C1RO9M 9887568 IC50 > 10000 nM T87670 C73TBN 10468802 IC50 >= 10000 nM T87670 C8LF3D 10858553 IC50 > 10000 nM T87670 C3TC7H 10871668 EC50 > 10000 nM T87670 CSG5H6 10902223 IC50 > 10000 nM T87670 CCI2L6 11045217 IC50 = 6910 nM T87670 CI8A6B 11076506 IC50 > 10000 nM T87670 C9E2AP 11152300 IC50 > 10000 nM T87670 C92AOP 11187538 IC50 > 10000 nM T87670 CYE8Q0 11244542 IC50 > 10000 nM T87670 CVH2C4 11321422 IC50 > 10000 nM T87670 CT8G0R 11338511 EC50 = 10700 nM T87670 CB26AX 11391631 IC50 > 10000 nM T87670 CFT60D 11475997 IC50 > 10000 nM T87670 C3L6FB 11748721 IC50 = 9770 nM T87670 C2FVO0 11830207 IC50 > 10000 nM T87670 CKG9Q1 12232068 IC50 > 10000 nM T87670 C5RJ6P 13045465 IC50 > 10000 nM T87670 C9CAK4 13166820 IC50 > 10000 nM T87670 CC5Q7O 14417955 IC50 > 10000 nM T87670 C0XNF5 14417956 IC50 = 10000 nM T87670 C9C0DT 14898643 IC50 > 10000 nM T87670 C5RCD3 14898644 IC50 > 10000 nM T87670 C7Q8HG 14950683 IC50 > 10000 nM T87670 CG49IS 14950684 IC50 > 10000 nM T87670 CLK42M 14950685 IC50 > 10000 nM T87670 CD13NW 14950686 IC50 > 10000 nM T87670 C39MRN 15262805 IC50 > 10000 nM T87670 CIJM09 16067243 IC50 > 10000 nM T87670 CV2QE8 16067244 IC50 > 10000 nM T87670 CM9XK7 16067272 IC50 > 10000 nM T87670 CZ7E3U 16067273 IC50 = 3450 nM T87670 C9Q7ZA 17171018 EC50 = 2 nM T87670 CTL0C7 21858022 IC50 > 10000 nM T87670 CF2S3C 21858023 IC50 > 10000 nM T87670 C4FED5 23612554 IC50 = 12000 nM T87670 C8RO1Q 23612567 IC50 = 640 nM T87670 CGN80J 23643046 IC50 > 10000 nM T87670 C8CU9Z 28640056 EC50 > 10000 nM T87670 CW4DJ1 44592049 IC50 = 10000 nM T87670 CIB17U 44592050 IC50 > 10000 nM T87670 C0PLI4 44592051 IC50 > 10000 nM T87670 CN91XU 44806719 IC50 > 10000 nM T87670 C0BQ4U 49890666 EC50 > 10000 nM T87670 C0YH3T 70677671 IC50 = 1770 nM T87670 CQT54O 70677672 IC50 = 10000 nM T87670 CR71AY 70677673 IC50 = 3990 nM T87670 C8VQ0M 70677674 IC50 > 10000 nM T87670 CURQ38 70677675 IC50 > 10000 nM T87670 CFMD45 70677677 IC50 = 3230 nM T87670 C2E1AD 70677804 IC50 = 10600 nM T87670 CVX9I7 70677805 IC50 > 10000 nM T87670 CLWV92 70677806 IC50 > 10000 nM T87670 CCE2U9 70677807 IC50 = 5080 nM T87670 C74KDW 70677808 IC50 > 10000 nM T87670 CK4C2I 70677809 IC50 > 10000 nM T87670 CTYE29 70677810 IC50 > 10000 nM T87670 CSGH58 70677953 IC50 = 6350 nM T87670 CY3O0R 70677954 IC50 > 10000 nM T87670 CCUW05 70677955 IC50 = 9000 nM T87670 CB4P6Y 70677956 IC50 > 10000 nM T87670 C6ESV8 70677957 IC50 > 10000 nM T87670 C3F2AY 70677958 IC50 > 10000 nM T87670 CV7Q3G 70677959 IC50 = 10000 nM T87670 C4Y1LE 70678097 IC50 = 358 nM T87670 C3DX1U 70678098 IC50 > 10000 nM T87670 C71DQG 70678099 IC50 = 261 nM T87670 CJ0P4V 70678100 IC50 > 10000 nM T87670 C82PMZ 70678101 IC50 = 113 nM T87670 CTB19O 70678102 IC50 > 10000 nM T87670 C46QGZ 70678238 IC50 = 854 nM T87670 CBX9D4 70678239 IC50 > 10000 nM T87670 CS7FL4 70678240 IC50 = 961 nM T87670 C30LIP 70678241 IC50 > 10000 nM T87670 CT1EF6 70678242 IC50 > 10000 nM T87670 CS6GV8 71581135 EC50 = 2.82 nM T87670 CDJH76 71682490 IC50 = 7140 nM T87670 C48BSN 71682637 IC50 = 5700 nM T87670 C1TAF4 71682638 IC50 > 10000 nM T87670 C0O9HE 71682639 IC50 = 981 nM T87670 CZE6R2 71682640 IC50 = 12800 nM T87670 C2FBL9 71682641 IC50 = 9320 nM T87670 CTOL05 71682642 IC50 = 13500 nM T87670 CDX59H 71682795 IC50 = 10300 nM T87670 C3S1OE 71682796 IC50 = 7690 nM T87670 CNM1Y8 71682797 IC50 = 5160 nM T87670 CJ3XH0 71682798 IC50 > 10000 nM T87670 C0HS4I 71682799 IC50 = 3290 nM T87670 C86ISD 71682800 IC50 = 10000 nM T87670 CK0Y3J 71682950 IC50 = 3760 nM T87670 C31ANM 71733843 IC50 = 21700 nM T87670 CU32CA 71733848 IC50 = 21700 nM T87670 CM7GX1 71733939 IC50 = 8920 nM T87670 CG8JP7 71733940 IC50 = 6200 nM T87670 CRMI92 71734946 IC50 = 29100 nM T87670 CUF29Z 73353471 EC50 = 1000 nM T87670 CO4IL2 76317959 IC50 > 10000 nM T87670 C5GI9Z 76325292 IC50 > 10000 nM T87670 CQE10H 85468767 IC50 = 3150 nM T87670 CA0Y8G 85469571 IC50 > 10000 nM T87670 CVY83X 90667465 IC50 > 10000 nM T87670 C85BUR 90667466 IC50 = 5560 nM T87670 C0FZU2 90667467 IC50 = 3460 nM T87670 C4MF8A 90667653 IC50 = 16400 nM T87670 CR2WI4 90667654 IC50 > 10000 nM T87670 C8N0LA 90667655 IC50 >= 10000 nM T87670 CU23VX 90667656 IC50 > 10000 nM T87670 CR8I5E 90667657 IC50 = 11800 nM T87670 CI61LD 90667658 IC50 > 10000 nM T87670 C7P2EG 90667659 IC50 > 10000 nM T87670 CS5DZ4 90667660 IC50 > 10000 nM T87670 C31ZMH 90667661 IC50 > 10000 nM T87670 CT37YL 90667662 IC50 >= 10000 nM T87670 CJ7V0Y 90667663 IC50 > 10000 nM T87670 C54BTS 90667664 EC50 = 1000 nM T87670 CJP21Z 90667665 IC50 = 6760 nM T87670 C9RM7U 90667666 IC50 > 10000 nM T87670 C18JNK 127029837 EC50 = 8.67 nM T87670 CZX4C2 127029838 EC50 = 0.69 nM T87670 C3L8GO 127030160 EC50 = 1.28 nM T87670 C3I4CH 127030161 EC50 = 0.4 nM T87670 C94VFD 127030831 IC50 = 7000 nM T87670 C74OQM 127031142 IC50 = 420 nM T87670 CYF8R3 127032327 IC50 = 770 nM T87670 C0VXZ2 127032328 IC50 = 2500 nM T87670 CMD50E 127032329 IC50 = 1800 nM T87670 CDFJ81 127033483 EC50 = 27.7 nM T87670 CXG07N 127033786 EC50 = 31.5 nM T87670 CB9OZ6 127034064 EC50 = 6.36 nM T87670 C30BCV 127034066 EC50 = 30.4 nM T87670 CK57OG 127034067 EC50 = 27.3 nM T87670 C4K9RW 127034068 EC50 = 19.6 nM T87670 CEH0S2 127034069 EC50 = 0.88 nM T87670 CSK5Y7 127034071 EC50 = 0.6 nM T87670 C36TFY 127034072 EC50 = 29.3 nM T87670 C6GPQ0 127034073 EC50 = 0.51 nM T87670 C9O7SI 127037894 EC50 = 12.4 nM T87670 C0KVN3 127037895 EC50 = 7.7 nM T87670 C30WOD 127038593 EC50 > 10000 nM T87670 CVJH84 127038962 EC50 = 30.9 nM T87670 C3MUN2 127042818 EC50 = 2 nM T87670 CLY3V5 137632605 EC50 = 500 nM T87670 CON1U3 137635440 EC50 > 30000 nM T87670 CQDA26 137635964 EC50 = 500 nM T87670 CU3HN7 137636853 EC50 > 30000 nM T87670 CV6E4P 137637218 EC50 = 300 nM T87670 CR21DQ 137639721 EC50 = 900 nM T87670 CHTK35 137640974 EC50 = 2000 nM T87670 CBO3M4 137641698 EC50 > 30000 nM T87670 C31DEB 137641866 EC50 > 30000 nM T87670 CRB6D0 137645195 EC50 = 500 nM T87670 C9DV0P 137648099 EC50 = 4000 nM T87670 CC7JM9 137648668 EC50 = 600 nM T87670 CG7YO2 137650491 EC50 = 20000 nM T87670 C52UVL 137651235 EC50 = 6000 nM T87670 C4R8IN 137654236 EC50 = 2000 nM T87670 CPF21A 137655056 EC50 = 200 nM T87670 C6O5AU 137655357 EC50 = 700 nM T87670 CXB65S 137658912 EC50 = 100 nM T87670 CP5S0R 137660243 EC50 = 1000 nM T87670 CSU48W 137661871 EC50 = 300 nM T87670 CP4YO0 142635551 EC50 = 1600 nM T87670 CR7FM4 145949041 EC50 = 20.24 nM T87670 C1F0BP 145949413 EC50 > 10000 nM T87670 CBC13V 145949551 EC50 > 10000 nM T87670 CXRO20 145950071 EC50 > 10000 nM T87670 CY60SW 145951064 IC50 = 2910 nM T87670 CCKN03 145951123 EC50 > 10000 nM T87670 CSG0W9 145951227 IC50 > 10000 nM T87670 C4LX7H 145951404 IC50 = 9450 nM T87670 C3G5TZ 145952824 IC50 = 6040 nM T87670 CS10GA 145953541 IC50 > 10000 nM T87670 CDI42H 145953879 IC50 > 10000 nM T87670 C6QX5T 145954189 EC50 > 10000 nM T87670 CKO9B4 145954190 EC50 > 10000 nM T87670 COMQ03 145954409 IC50 > 10000 nM T87670 C03WAH 145954816 EC50 > 10000 nM T87670 CUE8Y2 145955444 EC50 > 10000 nM T87670 CX95DH 145955833 EC50 > 10000 nM T87670 CG16ZX 145956544 IC50 = 3410 nM T87670 CA30EJ 145956612 IC50 > 10000 nM T87670 CW3A0Y 145958034 IC50 > 10000 nM T87670 CIK3B7 145958405 EC50 > 10000 nM T87670 CC5B9Y 145958428 IC50 > 10000 nM T87670 C3IH1U 145958480 IC50 > 10000 nM T87670 COP8M1 145958551 EC50 > 10000 nM T87670 CEQ9W7 145958588 EC50 > 10000 nM T87670 C5K9TY 145959141 IC50 = 4220 nM T87670 C25WFH 145960085 IC50 = 29300 nM T87670 CQ3B6P 145960178 IC50 = 10100 nM T87670 C5T2WE 145971274 EC50 > 10000 nM T87670 C6XAW4 145971463 EC50 > 10000 nM T87670 C4G8WI 145974549 IC50 = 3770 nM T87670 CFME69 155522092 EC50 > 10000 nM T87670 CB4FZ0 155527237 EC50 > 10000 nM T87670 C4XUO1 155527734 EC50 > 20000 nM T87670 C0Q8IM 155534990 EC50 > 10000 nM T87670 CEFS64 155566314 EC50 > 20000 nM T87670 D01RWS 16066912 IC50 = 5330 nM T87670 D01ZHW 5283389 IC50 > 10000 nM T87670 D02SMK 1172084 EC50 = 160 nM T87670 D08MON 16067266 IC50 = 6740 nM T87670 D08YQT 2125 EC50 = 630 nM T87670 D0B9RI 16067269 IC50 > 10000 nM T87670 D0D6OH 104895 EC50 = 1610 nM T87670 D0G3TV 2440433 EC50 = 260 nM T87670 D0G6BG 10731937 IC50 = 2810 nM T87670 D0Q9GU 1792197 EC50 = 110 nM T87670 D0R1ZD 59822766 EC50 = 158 nM T87670 D0UD9H 4302962 EC50 = 13600 nM T87670 D0Z0KY 11855860 EC50 = 316 nM T94692 CTJ3G2 9929785 EC50 = 1700 nM T94692 CL1O7Z 10500000 EC50 = 7000 nM T94692 CCO8I7 10500851 EC50 = 4000 nM T94692 C6B5CO 10525967 EC50 = 700 nM T94692 C5EHW0 10574243 EC50 = 2500 nM T94692 CX0ER5 10594954 EC50 = 2000 nM T94692 CCI8B6 10618856 EC50 = 1200 nM T94692 CWDB40 10689961 EC50 = 1300 nM T94692 C8WSP3 10691144 EC50 = 3800 nM T94692 CF0XW7 10714806 EC50 = 2000 nM T94692 CI1PM7 10715652 EC50 = 7600 nM T94692 C7Q6SJ 10761288 EC50 = 2000 nM T94692 C1E5BO 10786035 EC50 = 2000 nM T94692 C8FQ3T 10809488 EC50 = 1300 nM T94692 CM3TN5 11793747 EC50 = 1000 nM T94692 CAB3W9 11793994 EC50 = 700 nM T94692 C26HSZ 44341369 EC50 = 600 nM T00933 D0L5WM 2157 IC50 = 252000 nM T00933 D09NCT 53392492 IC50 = 10000 nM T00933 CWJ0U1 5312 IC50 = 2300 nM T00933 C06WZQ 222878 IC50 = 480 nM T00933 COS62U 245007 IC50 > 100000 nM T00933 C0MHV8 252439 IC50 = 1700 nM T00933 C2OS3W 2238068 IC50 = 117000 nM T00933 C2DBN5 46899607 IC50 = 19000 nM T00933 C2HXA1 53380104 IC50 = 58000 nM T00933 CMR1X3 56684140 IC50 > 1000000 nM T00933 CE26XI 56684141 IC50 > 1000000 nM T00933 CL8N7V 56964909 IC50 > 1000000 nM T00933 CLZ7P4 70702119 IC50 = 307000 nM T00933 CW1GP2 70702121 IC50 = 390000 nM T00933 CL3HT1 71449736 IC50 = 6900 nM T00933 CJH86V 71451542 IC50 = 11500 nM T00933 CH38AO 71453382 IC50 = 35000 nM T00933 C2U4AQ 71458738 IC50 = 3400 nM T00933 C14GIV 71735687 IC50 = 17000 nM T00933 CM02VN 71735839 IC50 = 14000 nM T00933 C4WS1H 71735840 IC50 = 23000 nM T00933 CT4YO5 71735841 IC50 = 43000 nM T00933 C2ZFM8 71735842 IC50 = 9100 nM T00933 CI5W0K 71735843 IC50 = 1200 nM T00933 CFY18G 73333510 IC50 = 150000 nM T00933 CN5B4O 73352277 IC50 = 24000 nM T00933 CMR52S 78426698 IC50 = 7700 nM T00933 CQY0K3 91938043 IC50 < 250 nM T00933 C2S1AO 110264830 IC50 > 25000 nM T00933 CPSD31 118420829 IC50 < 250 nM T00933 CH6FX3 118421371 IC50 < 250 nM T00933 C6YT2Q 118598059 IC50 > 4000 nM T00933 CJVK69 119081409 IC50 > 25000 nM T00933 C5IZD1 122181577 IC50 > 100000 nM T00933 CRM93S 122181583 IC50 > 100000 nM T00933 CU57QX 122181584 IC50 = 73000 nM T00933 C9QVZ5 122181587 IC50 = 29000 nM T00933 CJQ91K 122181588 IC50 = 24000 nM T00933 CIJ0G6 127030272 IC50 < 250 nM T00933 C2EY1K 127033166 IC50 < 250 nM T00933 CID1E9 127034046 IC50 < 250 nM T00933 C4QC5Y 145960532 IC50 = 242000 nM T00933 C8HPT2 145961258 IC50 = 496000 nM T00933 C9FGU1 145961684 IC50 = 126000 nM T00933 CF4ME6 145962269 IC50 = 355000 nM T00933 CZP8B7 145962316 IC50 = 1700 nM T00933 CJGC76 145962553 IC50 = 397000 nM T00933 CK3DZ7 145962837 IC50 = 286000 nM T00933 CVU6M3 145962898 IC50 = 240000 nM T00933 C3RB8P 145963156 IC50 = 386000 nM T00933 CK96HI 145963214 IC50 = 377000 nM T00933 C81CRJ 145963620 IC50 = 221000 nM T00933 C2WKX0 145963644 IC50 = 697000 nM T00933 CIM7D4 155548682 IC50 > 50000 nM T00933 CFR06L 155551969 IC50 > 50000 nM T00933 D07IOY 10365 IC50 > 250000 nM T00933 D08IZY 3080614 IC50 > 250000 nM T00933 D0B2WZ 15331 IC50 = 550 nM T44684 CW68DS 71542548 IC50 = 3 nM T44684 C4Z9NE 71712019 IC50 = 4 nM T44684 C9W2QU 73441909 IC50 = 1 nM T44684 C37AFR 73441957 IC50 = 3 nM T44684 CLO08N 118732177 IC50 = 3 nM T44684 CLJ5Q3 118732178 IC50 = 1 nM T44684 CBUT48 118732179 IC50 = 24 nM T44684 CTD5J0 118732180 IC50 = 656 nM T44684 CE4PC8 118732181 IC50 = 161 nM T44684 C7VA3N 118732182 IC50 = 29 nM T44684 CD2U5R 118732183 IC50 = 119 nM T44684 CY1ES6 118732184 IC50 = 62 nM T44684 CE7MX2 118732185 IC50 = 1 nM T44684 C64ACS 118732186 IC50 = 2 nM T44684 C6MUQ2 118732187 IC50 = 4 nM T44684 CH4YL5 118732188 IC50 = 2241 nM T44684 CEGM19 118732189 IC50 = 6 nM T44684 C4WY7T 118732190 IC50 = 2 nM T44684 CKE83Y 118732191 IC50 = 1 nM T44684 CWC0U9 118732192 IC50 = 2 nM T97613 D0AN7B 896 EC50 = 0.0257 nM T97613 D0T7OW 681 Ki = 7100 nM T97613 D0U0KW 208902 Ki = 0.0138 nM T97613 D0D8FN 219018 Ki = 0.07943 nM T97613 D01ESJ 122162 Ki = 158 nM T97613 D0Y8UB 82148 Ki = 0.06 nM T97613 CHA7C3 12111 EC50 = 237000 nM T97613 C1XYC4 34247 IC50 = 1.259 nM T97613 CSU58J 164405 IC50 = 1.259 nM T97613 CZ3LQ4 189748 Ki = 207 nM T97613 CY8NS0 320362 Ki = 5200 nM T97613 CYVK43 588712 IC50 = 6309.57 nM T97613 C59MGT 594980 IC50 = 0.7943 nM T97613 C72CAB 1550607 Ki = 1900 nM T97613 CRZ4O6 2368416 IC50 = 3981.07 nM T97613 C1BV0A 2821758 IC50 = 1995.26 nM T97613 CJY81E 3071630 IC50 = 2.512 nM T97613 CJ5AE2 3071631 IC50 = 1.995 nM T97613 C03HMX 3071635 IC50 = 100 nM T97613 C2S0HM 3071647 IC50 = 2511.89 nM T97613 C3HJK8 3525815 EC50 = 920 nM T97613 COT3G9 3956219 Ki = 14.6 nM T97613 CJPD17 3964826 Ki = 61659.5 nM T97613 CK8RT4 4207624 Ki = 37153.52 nM T97613 CX0OC9 5151463 Ki = 4168.69 nM T97613 C8CM9B 9795837 Ki > 500 nM T97613 CXW4G5 9796251 Ki = 2.08 nM T97613 CI2A3Y 9796846 Ki = 0.012 nM T97613 C59VTY 9797460 Ki = 0.016 nM T97613 C7VG4A 9797715 Ki > 500 nM T97613 CB79WC 9798080 Ki = 0.057 nM T97613 C41QXC 9805364 Ki = 2.05 nM T97613 CWG0C2 9817006 IC50 = 77.6 nM T97613 CIL4T9 9817262 Ki = 0.19 nM T97613 C3ND5E 9817636 Ki = 0.95 nM T97613 CD3YQ2 9817692 Ki > 500 nM T97613 C89NSW 9818487 Ki = 53 nM T97613 CC0GV2 9819843 Ki = 31.5 nM T97613 C76BTA 9834952 IC50 = 1 nM T97613 C80PNI 9837740 IC50 = 7.943 nM T97613 C9Q0SO 9837777 IC50 = 501.19 nM T97613 C6K8DF 9839199 Ki = 0.11 nM T97613 CGO7V4 9839629 Ki = 0.01 nM T97613 C78CMN 9840277 Ki = 0.026 nM T97613 CDWY16 9840647 Ki = 4.37 nM T97613 C3NU4X 9850873 EC50 > 0.00001 nM T97613 CK8YO6 9858255 Ki = 1.82 nM T97613 C43NXF 9859693 Ki = 786 nM T97613 C2ENY0 9859913 Ki = 84 nM T97613 CXO8S2 9859969 IC50 = 0.875 nM T97613 CM0LY6 9860296 Ki = 3.9 nM T97613 CB0R8G 9860588 Ki = 8.9 nM T97613 CO12LY 9860638 Ki > 500 nM T97613 C05WRO 9861677 IC50 = 3880 nM T97613 CT5XP8 9870683 Ki = 1.38 nM T97613 CD9LZ7 9873402 Ki = 0.03 nM T97613 C38VXA 9881916 IC50 = 5.012 nM T97613 C5LQ7P 9881917 Ki = 300 nM T97613 C7X3QW 9883864 Ki = 0.07 nM T97613 CG1ID3 9884156 Ki = 53.7 nM T97613 C1IBZ4 9884406 Ki = 0.75 nM T97613 CT93HK 9888609 Ki = 5.2 nM T97613 CVR15A 9893513 Ki = 0.08 nM T97613 CO3JD2 9903515 Ki = 0.01 nM T97613 CV1CX0 9903953 Ki > 500 nM T97613 C4U7DC 9904304 Ki = 0.008 nM T97613 C8FVR1 9909783 Ki < 1000 nM T97613 C2O3FD 9914839 Ki = 0.05 nM T97613 C9WSM4 9916005 Ki = 0.05 nM T97613 CCUJ86 9925797 Ki = 0.1 nM T97613 CUQ86C 9925874 Ki > 500 nM T97613 CZJP28 9926304 Ki = 0.015 nM T97613 C6MEF3 9927219 IC50 = 0.01585 nM T97613 C3VE1W 9930390 Ki = 84.5 nM T97613 C0CGA4 9937825 Ki = 0.92 nM T97613 CFG16W 9947753 Ki = 63 nM T97613 C9SAE0 9948714 Ki = 0.2 nM T97613 C2YJC7 9970584 Ki = 8.1 nM T97613 CDC41T 9975634 IC50 = 1.259 nM T97613 CNM4S1 9993398 IC50 = 10 nM T97613 C1P8AI 9998754 Ki = 0.05 nM T97613 CYT93Z 10015474 Ki = 3 nM T97613 CWT07A 10015475 Ki = 3.5 nM T97613 CM52OT 10016733 Ki = 0.05 nM T97613 CHW0S6 10016919 Ki = 0.099 nM T97613 C3W4AZ 10019103 Ki = 1.288 nM T97613 CDZ71M 10022490 Ki = 3.7 nM T97613 C8JRV7 10022570 Ki = 1.3 nM T97613 CB8XI1 10038243 Ki = 2.3 nM T97613 C79HTQ 10038961 IC50 = 10 nM T97613 C8NSX9 10039072 IC50 = 19.95 nM T97613 C05RQN 10044270 Ki = 797 nM T97613 C72AIR 10059969 IC50 = 15.85 nM T97613 C9TAU5 10060719 IC50 = 158.49 nM T97613 C04FNQ 10061064 Ki = 6.9 nM T97613 C0Z3NI 10061999 IC50 = 1.995 nM T97613 CT03BO 10069719 Ki = 19.2 nM T97613 C9LNC0 10085672 IC50 = 501.19 nM T97613 CGO3N1 10089253 Ki = 1.3 nM T97613 CX57TO 10091075 Ki = 3.3 nM T97613 C7NE5J 10131203 IC50 = 10 nM T97613 CKC1Y7 10163052 Ki = 0.09 nM T97613 C0IP4U 10198772 IC50 > 10000 nM T97613 CZ5I7D 10199282 Ki = 0.8 nM T97613 CJF79Z 10243074 IC50 = 3162.28 nM T97613 C2PXR8 10245336 Ki = 199.53 nM T97613 C0X3VG 10248871 IC50 = 5.012 nM T97613 C9DSM8 10265261 IC50 = 1 nM T97613 CC7T3G 10265421 IC50 = 6.31 nM T97613 C7CLE4 10266979 IC50 = 200 nM T97613 C0HJ7G 10301190 Ki = 2.37 nM T97613 CZQE69 10332159 Ki = 2.8 nM T97613 C4Z6QS 10333442 Ki = 2.2 nM T97613 C1LVM8 10333620 IC50 = 3.981 nM T97613 CGSO61 10361427 Ki = 0.76 nM T97613 C9I7ML 10377971 IC50 = 19.95 nM T97613 C3ELV5 10379422 IC50 = 39.81 nM T97613 CS5LV2 10384120 Ki = 7.5 nM T97613 CM8WL2 10385056 Ki = 21.6 nM T97613 C3VU0Z 10390683 Ki = 93 nM T97613 C9C8HL 10399169 IC50 = 125.89 nM T97613 C9KLP2 10399579 Ki = 5.9 nM T97613 CJ4D8T 10400294 Ki = 0.7 nM T97613 CM23IA 10422677 IC50 = 5.012 nM T97613 C8HKY5 10423378 Ki = 0.05 nM T97613 C9ND1W 10424693 Ki = 5 nM T97613 CEZ75R 10427851 Ki = 1390 nM T97613 C8Y7JV 10428383 Ki = 1288.25 nM T97613 C5Z9GU 10446712 Ki = 0.05 nM T97613 COA8E4 10447987 Ki = 181.97 nM T97613 CPZ68G 10448305 IC50 = 19.95 nM T97613 C1ZN2H 10452167 Ki = 0.05 nM T97613 CSUN05 10454621 Ki = 1880 nM T97613 C0Y1UP 10465460 Ki = 2454.71 nM T97613 C7L8GS 10468642 Ki = 0.65 nM T97613 C32SXQ 10495702 Ki = 4.3 nM T97613 CK4P3O 10513751 Ki = 630.96 nM T97613 C6BIK5 10513752 Ki = 16218.1 nM T97613 CCM6O4 10515048 Ki = 0.79 nM T97613 CB6QE5 10517621 Ki = 195 nM T97613 C2VEM4 10518621 Ki = 204 nM T97613 CJ9K8Z 10518884 Ki = 87.1 nM T97613 C0YLB4 10520058 Ki = 282 nM T97613 CIR20T 10522674 Ki = 8.91 nM T97613 CVB47I 10522675 Ki = 4.07 nM T97613 C85RBH 10526493 Ki = 100 nM T97613 CJF51I 10540964 Ki = 0.22 nM T97613 CW1X2B 10542922 Ki = 1.89 nM T97613 CG9VZ2 10544425 Ki = 1200 nM T97613 C4B2CY 10545399 Ki = 42 nM T97613 CQ3M0U 10561982 Ki = 2.65 nM T97613 CJ6W3C 10562968 Ki = 0.12 nM T97613 CXV4U3 10563168 Ki = 524.81 nM T97613 C8FR1M 10567427 Ki = 776 nM T97613 CXW7T3 10567865 Ki = 63.1 nM T97613 CSR1Q3 10591657 Ki = 174 nM T97613 C6N2VC 10595585 Ki = 437 nM T97613 C6H7DI 10596576 Ki = 257 nM T97613 CC9YR3 10609620 Ki = 8511.38 nM T97613 CX6NI4 10610443 Ki = 134.9 nM T97613 C0Y8VE 10611901 Ki = 6.41 nM T97613 CQ0MA7 10616723 Ki = 7.24 nM T97613 C10KPW 10617720 Ki = 14.5 nM T97613 COE89Y 10620323 Ki = 2950 nM T97613 COZ28S 10637638 Ki = 10 nM T97613 C59HRX 10638747 Ki = 3981.07 nM T97613 C6M5VE 10639585 Ki = 630.96 nM T97613 C2I6TL 10640625 Ki = 831.76 nM T97613 C2L9MR 10640828 Ki = 0.66 nM T97613 CJZ06I 10641756 Ki = 288 nM T97613 CJK2Z3 10656443 Ki = 1230.27 nM T97613 C9OI8Y 10657206 Ki = 407.38 nM T97613 CFJ95P 10658090 Ki = 2951.21 nM T97613 CQ30BW 10659603 Ki = 0.1 nM T97613 CCTW96 10661735 Ki = 0.37 nM T97613 CC0G7X 10663827 IC50 > 1000 nM T97613 CZE91U 10664333 Ki = 115 nM T97613 C1U4EO 10666373 Ki = 513 nM T97613 C04IND 10704399 Ki = 4.24 nM T97613 CEK93Y 10704742 Ki = 3801.89 nM T97613 C38JKD 10705590 Ki = 1819.7 nM T97613 CNS05E 10709646 Ki = 389 nM T97613 CHE67R 10711649 Ki = 70.8 nM T97613 CB7CD3 10712600 Ki = 46.8 nM T97613 CHUL45 10712733 Ki = 5.89 nM T97613 CY3PD6 10714573 Ki = 269 nM T97613 CD27QT 10729569 Ki = 4.34 nM T97613 CW6XT7 10736247 Ki = 2040 nM T97613 C0FN2D 10737123 Ki = 251 nM T97613 CM6K0U 10737372 Ki = 52.5 nM T97613 C27XEV 10738183 Ki = 501 nM T97613 CO2WK7 10752506 Ki = 1.2 nM T97613 CWNB23 10753255 Ki = 1.06 nM T97613 CZJL23 10754723 Ki = 2.2 nM T97613 CC7XK5 10760155 Ki = 275 nM T97613 C6Q0YV 10763177 Ki = 1.3 nM T97613 C17NJY 10778397 Ki = 0.41 nM T97613 CATC31 10800029 Ki = 6.5 nM T97613 C15GYJ 10801655 Ki = 6.48 nM T97613 CP87NG 10807560 Ki = 79.4 nM T97613 CU3YN6 10808489 Ki = 234 nM T97613 CNM36T 10829695 Ki = 141.25 nM T97613 CRQJ04 10831675 Ki = 11 nM T97613 C74HBT 10850411 Ki = 1.32 nM T97613 CG74JD 10853020 Ki = 148 nM T97613 C2RE6J 10853021 Ki = 240 nM T97613 CT0S8G 10854190 Ki = 18.2 nM T97613 CQZ4J3 10873443 Ki = 1.1 nM T97613 C4LX0I 10882307 Ki = 5.37 nM T97613 C1O5HT 10893437 Ki = 691.83 nM T97613 CS1O3P 10903368 Ki = 1288.25 nM T97613 CTS64X 10903463 Ki = 50.12 nM T97613 CQV6L3 10925379 Ki = 0.04 nM T97613 C47ROS 10925526 Ki = 66.4 nM T97613 CFZ13L 10925712 Ki = 0.01 nM T97613 C6S3NQ 10926138 Ki = 3.51 nM T97613 C7PYU9 10938056 Ki = 8.2 nM T97613 CJ52CX 10946222 Ki = 8560 nM T97613 C0B4CW 10948786 Ki = 698 nM T97613 CXK4T2 10950593 Ki = 476 nM T97613 C6LKR7 10956792 Ki = 1060 nM T97613 C7DMI9 10959837 Ki = 42.7 nM T97613 C3MU2F 10969292 Ki = 64.4 nM T97613 CAJ30W 10991315 Ki = 309.03 nM T97613 C6GJ3W 11002150 Ki = 331.13 nM T97613 CDO6V1 11002840 Ki = 7.19 nM T97613 C3YNE2 11014883 Ki = 239.88 nM T97613 C0UB2R 11045144 Ki = 275.42 nM T97613 CW7M5P 11046748 Ki = 55 nM T97613 C9FQH2 11058163 Ki = 3162.28 nM T97613 CFJG64 11059058 IC50 = 1740 nM T97613 C7EAI8 11065731 Ki = 49 nM T97613 CCW92A 11066802 Ki = 223.87 nM T97613 C0J9PL 11068422 Ki = 12.9 nM T97613 CEJZ12 11078652 Ki = 288 nM T97613 C8KO9X 11079938 Ki = 0.3 nM T97613 C6RL3D 11088627 Ki = 29 nM T97613 CX04WH 11098363 Ki = 155 nM T97613 C9R2PL 11100761 Ki = 0.08 nM T97613 CKT2U4 11109646 Ki = 569 nM T97613 CNS0V2 11110447 Ki = 1.01 nM T97613 CS1YX7 11131123 Ki = 229 nM T97613 C0CSN9 11165283 Ki = 9 nM T97613 C1Q4HG 11173131 Ki = 239.88 nM T97613 C8YVE2 11178762 IC50 = 230 nM T97613 C2C6WP 11208578 Ki = 20417.38 nM T97613 CS9ZN3 11208632 Ki = 549.54 nM T97613 CY9NP7 11213541 IC50 > 1000 nM T97613 CSQB21 11219713 Ki = 389.05 nM T97613 C2U4IR 11247050 IC50 > 1000 nM T97613 CK17JA 11277044 Ki = 549.54 nM T97613 CLXE76 11287002 Ki = 20892.96 nM T97613 CCND09 11304958 IC50 > 1000 nM T97613 CUM40C 11304981 IC50 > 1000 nM T97613 CM2EL5 11310062 Ki = 63095.73 nM T97613 C9D2WI 11314110 Ki < 10000 nM T97613 CQ9ZV4 11326232 Ki < 10000 nM T97613 C8VX2J 11351216 Ki = 22.1 nM T97613 C03UAY 11361621 IC50 = 621 nM T97613 CT15EV 11392720 Ki = 162.18 nM T97613 C2CT0K 11393103 Ki = 57.54 nM T97613 CF20YO 11403195 Ki = 112.2 nM T97613 C31TXA 11418246 Ki = 915 nM T97613 CUE25A 11426853 Ki = 3.02 nM T97613 CF8E2S 11430378 IC50 = 673 nM T97613 C9PW1B 11463056 Ki = 226 nM T97613 C12YKO 11476283 IC50 > 1000 nM T97613 CDXY43 11485537 Ki < 10000 nM T97613 C2F8XC 11500596 Ki = 493 nM T97613 COR3H7 11501012 Ki = 479 nM T97613 CS9KZ5 11507534 Ki = 6.03 nM T97613 C97PGC 11515177 Ki = 170 nM T97613 CN4WO8 11529521 Ki = 57.8 nM T97613 CKXL24 11536746 Ki = 148 nM T97613 CJP73K 11536939 Ki = 10.6 nM T97613 C45FJW 11543959 Ki = 116 nM T97613 C90FCS 11550834 Ki = 4.9 nM T97613 C9H5ND 11573203 Ki = 307 nM T97613 C4EOD5 11581340 Ki = 1 nM T97613 CU63XE 11587169 Ki = 11.5 nM T97613 CS5A0D 11595087 Ki = 589 nM T97613 CIQM18 11602301 Ki = 468 nM T97613 CMQ46D 11616029 Ki = 176 nM T97613 CE75OU 11616210 Ki = 483 nM T97613 C3T9BS 11623375 Ki = 86 nM T97613 C43EBC 11624018 Ki = 714 nM T97613 C0FTQ4 11637615 Ki = 8.2 nM T97613 C09NDO 11638009 Ki = 34 nM T97613 C9E1XH 11644612 Ki = 1.22 nM T97613 CNL3G5 11652196 Ki = 4.27 nM T97613 CAS86V 11666721 Ki = 1100 nM T97613 CD48BG 11680808 Ki = 65.7 nM T97613 C5YRT3 11681026 Ki = 8.51 nM T97613 C9EKN8 11681201 Ki = 302 nM T97613 C1CT0E 11688043 Ki = 212 nM T97613 C0LR6M 11702296 Ki = 28 nM T97613 CU6A7S 11723593 Ki = 0.02 nM T97613 C0MD4I 11733059 Ki = 8.67 nM T97613 CM4UF5 11741001 Ki = 0.05 nM T97613 C25BDQ 11749479 IC50 = 512 nM T97613 C8LYO7 11776674 Ki = 2.239 nM T97613 CI70SF 11784134 Ki = 80 nM T97613 C97WON 11784859 IC50 > 1000 nM T97613 CT49OP 11791741 Ki = 117 nM T97613 CH1YN6 11794657 Ki = 759 nM T97613 CDQ10E 11810280 Ki = 3.29 nM T97613 CI7SV5 11824364 Ki = 14.3 nM T97613 CRDE14 11824365 Ki = 24 nM T97613 CA5UO1 12004056 Ki = 1.445 nM T97613 C7X6FI 12071674 Ki = 4 nM T97613 C0X9NG 12288745 IC50 = 10000 nM T97613 C5TW9V 12436514 Ki = 12022.64 nM T97613 C3BJ6H 12436515 Ki = 1380.38 nM T97613 C5M9RC 12436516 Ki = 11481.54 nM T97613 C6AOC8 12985489 Ki = 5.9 nM T97613 C7IA6C 12985490 Ki = 297 nM T97613 CQS49L 12985491 Ki = 50.7 nM T97613 C24RNV 12985492 Ki = 126 nM T97613 C1SH0A 12985493 Ki = 204 nM T97613 CIP19Y 12985494 Ki = 125 nM T97613 CLB6Q2 12985495 Ki = 60.3 nM T97613 C8XT9Y 12985496 Ki = 1510 nM T97613 C4DFR8 13250272 Ki = 3801.89 nM T97613 CRXP16 15149133 IC50 = 1995.26 nM T97613 CFS15K 15149134 IC50 = 100000 nM T97613 C2E7TH 15289276 IC50 = 0.3162 nM T97613 CR6NI0 15289277 IC50 = 15.85 nM T97613 C4LSV3 15340628 IC50 = 158.49 nM T97613 COR35C 15340631 IC50 = 1.259 nM T97613 C5L8HX 15340632 IC50 = 0.1585 nM T97613 C74ASW 15340633 IC50 = 0.2512 nM T97613 C3R9KO 15372705 IC50 = 10000 nM T97613 C4SOP3 15372706 IC50 = 31622.78 nM T97613 C06KCV 15391785 IC50 = 15848.93 nM T97613 CQ19IZ 15391788 IC50 = 10000 nM T97613 C7QAE3 15391789 IC50 = 39.81 nM T97613 CP0SV7 15453084 Ki = 0.3 nM T97613 CHEF08 15453090 Ki = 0.06 nM T97613 C5B9CQ 15453093 Ki = 3.7 nM T97613 CTC6L1 15453819 Ki = 180 nM T97613 CY27AW 15453821 Ki = 29 nM T97613 CC9F6Z 15838838 IC50 = 10000 nM T97613 CZU2Q8 15838839 IC50 = 501.19 nM T97613 C9OB6C 15838841 IC50 = 7943.28 nM T97613 C6YB2V 16094576 Ki = 707.95 nM T97613 C46PJR 16094577 Ki = 524.81 nM T97613 C1SG9Y 16094578 Ki = 1202.26 nM T97613 CHG14X 16094579 Ki = 389.05 nM T97613 C3JUF7 16094580 Ki = 69.18 nM T97613 CE46TJ 16094582 Ki = 512.86 nM T97613 CJ2F5Y 16094583 Ki = 912.01 nM T97613 C6F4KQ 16094585 Ki = 93.33 nM T97613 C82AWU 16094586 Ki = 58.88 nM T97613 CF3S2Z 16094587 Ki = 363.08 nM T97613 CJR8Q3 16094588 Ki = 549.54 nM T97613 CIE61K 16094591 Ki = 691.83 nM T97613 C15SJU 16094592 Ki = 3630.78 nM T97613 CFLI78 16094593 Ki = 229.09 nM T97613 CY47EW 16094594 Ki = 257.04 nM T97613 C7MHQ5 16094595 Ki = 2187.76 nM T97613 CFR04C 16105169 Ki = 1000 nM T97613 CIV2T9 16105170 Ki = 1778.28 nM T97613 CU0DZ6 16656789 Ki = 4.169 nM T97613 C0QVE3 16743123 Ki = 75.86 nM T97613 C71WVP 16743124 Ki = 114.82 nM T97613 CTP8F7 16743125 Ki = 371.54 nM T97613 CF4L3D 16743288 Ki = 5888.44 nM T97613 CP30ZO 16743294 Ki = 190.55 nM T97613 C0SEN7 16743295 Ki = 41.69 nM T97613 C2BG5R 16743464 Ki = 2630.27 nM T97613 CGAW53 16750566 Ki = 7.91 nM T97613 CRG52N 16750569 Ki = 5.129 nM T97613 C87YMC 17524911 IC50 = 6309.57 nM T97613 CI19XZ 17956989 IC50 > 10000 nM T97613 CWC8V1 17957000 IC50 = 85.4 nM T97613 CXG63C 17957007 IC50 = 5350 nM T97613 CU83BG 18007928 EC50 = 3.14 nM T97613 C9O1UG 18007985 Ki = 1.07 nM T97613 CHLP82 18174996 IC50 > 10000 nM T97613 CZ2H3M 18175008 IC50 = 310 nM T97613 CAT5L1 18175018 IC50 = 10000 nM T97613 CE6YD4 18175028 IC50 = 5000 nM T97613 CX7D3G 18175032 IC50 = 2610 nM T97613 CAU40C 18175057 IC50 > 10000 nM T97613 C5FK7U 18177433 IC50 = 1000 nM T97613 CWP5C8 18177435 IC50 = 63.1 nM T97613 C5M3VT 18177465 IC50 = 794.33 nM T97613 CZT1C0 18357874 IC50 = 1000 nM T97613 C78NQP 18360631 Ki = 0.26 nM T97613 C0N4ZE 18360658 EC50 = 1.94 nM T97613 CVJ23S 18360745 IC50 = 2.512 nM T97613 C0DJM4 18466111 Ki = 0.03 nM T97613 C36XYE 18522208 Ki = 19 nM T97613 C2UZL1 18522267 Ki = 16 nM T97613 CE5Q1P 18522272 Ki = 6 nM T97613 C87AHP 18702059 Ki = 99 nM T97613 C3PC0I 18782997 IC50 = 1584.89 nM T97613 CFDM12 18783019 IC50 = 5.012 nM T97613 CSN8Z3 18783022 IC50 = 3.981 nM T97613 CP1HO6 18947270 IC50 = 79.43 nM T97613 CB2EZ8 18947294 IC50 = 3.162 nM T97613 C1DY6K 18947318 IC50 = 50.12 nM T97613 CL4F8W 18947325 IC50 = 7.943 nM T97613 C9YX2E 19086015 IC50 = 251.19 nM T97613 CYBN06 19385775 IC50 = 12.59 nM T97613 CNB5D9 19696845 IC50 = 12.59 nM T97613 C7FWI9 19703003 IC50 = 0.01259 nM T97613 CRO46J 19703015 Ki = 1.6 nM T97613 C4KJP0 19703028 IC50 = 1584.89 nM T97613 CD5FI1 19703043 IC50 = 2511.89 nM T97613 C61QAX 19703053 IC50 = 10000 nM T97613 C1I0OZ 19703063 Ki = 40 nM T97613 CVB5J6 19703067 IC50 = 10000 nM T97613 C09IUF 19752678 IC50 = 19.95 nM T97613 CQ3KE5 19967248 IC50 = 3.981 nM T97613 CS2VZ6 20355585 Ki = 1.34 nM T97613 CS5KB7 20590652 Ki = 2 nM T97613 C8KEI5 20590653 Ki = 1 nM T97613 CDXF27 20590654 Ki = 1 nM T97613 C6V1TU 20590664 Ki = 33 nM T97613 CNS15E 20590665 Ki = 6 nM T97613 CEM7F6 20642483 Ki = 1.2 nM T97613 CPVH03 21460931 IC50 = 1584.89 nM T97613 CX75WM 21469682 IC50 = 630.96 nM T97613 CY8XU0 21469690 IC50 = 100 nM T97613 CDY18E 21469691 IC50 = 63.1 nM T97613 CGX1R5 21469693 IC50 = 794.33 nM T97613 C6N7UG 21572387 IC50 = 501.19 nM T97613 CL64ZO 21581653 Ki = 9.5 nM T97613 C90HJK 21581654 Ki = 0.2 nM T97613 C6ZQD8 21916760 IC50 = 477 nM T97613 CZ2AW7 22004791 Ki = 0.045 nM T97613 CD6V5I 22004862 Ki = 0.0082 nM T97613 C1AX5C 22037991 IC50 > 1000 nM T97613 CASG07 22133298 IC50 = 50.12 nM T97613 CO4A0H 22375366 IC50 = 156 nM T97613 CO1L6H 22375370 IC50 > 1000 nM T97613 CVJX25 22375372 IC50 = 160 nM T97613 CU4T2X 22375392 IC50 > 1000 nM T97613 C90OUD 22375402 IC50 > 1000 nM T97613 CIE2B1 22375407 IC50 > 1000 nM T97613 C6CQ5D 22375417 IC50 > 1000 nM T97613 CELS26 22718521 Ki = 183 nM T97613 CS3WC4 22718530 Ki = 40 nM T97613 C5FD7I 22718548 Ki = 87 nM T97613 CS4IY9 22718555 Ki = 40 nM T97613 C7FX6M 22718571 Ki = 166 nM T97613 CZ6D9B 22718576 Ki = 24 nM T97613 CRQT08 22718579 Ki = 116 nM T97613 CR46PF 22718585 Ki = 142 nM T97613 C4XJ6L 22718596 Ki = 60 nM T97613 CM6ZG9 22718602 Ki = 13.2 nM T97613 CEC0I5 22718610 Ki = 13.1 nM T97613 CB2QJ0 22718619 Ki = 119 nM T97613 CR5D8T 22718654 Ki = 60 nM T97613 CSPB82 22718661 Ki = 51 nM T97613 CA4MY6 23360808 IC50 = 6.31 nM T97613 CBLN82 23360817 IC50 = 39.81 nM T97613 C14VPT 23360832 IC50 = 50.12 nM T97613 C4OC9V 23360842 IC50 = 7.943 nM T97613 CYHK42 23360848 IC50 = 15.85 nM T97613 CJY48G 23360853 IC50 = 125.89 nM T97613 CL4CF8 23642306 Ki = 1.349 nM T97613 C9U6TM 23642307 Ki = 4.677 nM T97613 CG78OH 23658143 Ki = 346.74 nM T97613 CY68EQ 23658144 Ki = 5.888 nM T97613 CBS59I 23658145 Ki = 181.97 nM T97613 CLJ03E 23658146 Ki = 3.388 nM T97613 C3X5PA 24750069 Ki = 50.12 nM T97613 CPLG20 24750070 Ki = 5.248 nM T97613 C6NQP2 24750071 Ki = 4.169 nM T97613 CUZ3C2 24750077 Ki = 19.05 nM T97613 C67HYD 24750188 Ki = 100 nM T97613 C51VEA 24750189 Ki = 131.83 nM T97613 CAV48F 24750190 Ki = 125.89 nM T97613 CQD54L 24750191 Ki = 16.98 nM T97613 CYQ6A7 24750193 Ki = 0.8318 nM T97613 CYFL67 24750194 Ki = 323.59 nM T97613 CO87FN 24750195 Ki = 1288.25 nM T97613 CK0AC4 24954990 Ki = 0.039 nM T97613 C8A5QN 24954991 Ki = 0.16 nM T97613 CZE7M2 24954992 Ki = 0.48 nM T97613 CRU4L6 24955342 Ki > 100 nM T97613 CQFI43 24955343 Ki = 0.082 nM T97613 CFPI79 25014882 IC50 = 8180 nM T97613 C21GCY 25022429 Ki = 9.8 nM T97613 C8K5GJ 25022442 Ki = 302 nM T97613 C6P0QW 25209860 Ki = 147.91 nM T97613 C8E9JX 25209861 Ki = 40.74 nM T97613 CLW71G 25209998 Ki = 5.754 nM T97613 CGSV97 25209999 Ki = 85 nM T97613 C4RPN9 25210000 Ki = 302 nM T97613 C7WY8N 25210131 Ki = 38 nM T97613 CFU8K9 25210132 Ki = 1400 nM T97613 C96ZPF 25210133 Ki = 40.74 nM T97613 C54OEZ 25210134 Ki = 120.23 nM T97613 CJQX17 25210135 Ki = 108 nM T97613 CM93GU 25270146 Ki = 3.7 nM T97613 CH15NX 39847023 Ki = 59000 nM T97613 CY1K7H 44241665 IC50 = 3.14 nM T97613 CRE65K 44241666 Ki = 15.49 nM T97613 CFB6X3 44264689 Ki = 61 nM T97613 CG8OF4 44264692 Ki > 500 nM T97613 C15DKZ 44264705 Ki = 31 nM T97613 CN0ZJ8 44264706 Ki = 61 nM T97613 C6Z7EG 44264707 Ki = 84 nM T97613 CUOG79 44264769 Ki = 1.1 nM T97613 CUSJ15 44264818 Ki = 10.9 nM T97613 C8K7XE 44264843 Ki = 34 nM T97613 CJNR68 44264844 Ki = 12 nM T97613 CI0PL7 44264849 Ki = 106 nM T97613 C6XF9C 44264857 Ki > 500 nM T97613 C1GKR5 44264861 Ki = 36 nM T97613 C5GKS4 44264871 Ki = 18 nM T97613 CJIZ29 44264892 Ki = 1 nM T97613 CCXI31 44264903 Ki = 0.05 nM T97613 CKV1H3 44264904 Ki = 41 nM T97613 CLQ9O0 44264909 Ki = 92 nM T97613 C5U1EH 44264942 Ki = 92 nM T97613 CJUS17 44264949 Ki = 63 nM T97613 C3HKR4 44264950 Ki > 500 nM T97613 CF82IP 44264962 Ki = 98 nM T97613 CNXG58 44264964 Ki > 500 nM T97613 C32BSH 44264965 Ki > 500 nM T97613 CP9SA3 44264982 Ki > 500 nM T97613 CF59MU 44264983 Ki > 500 nM T97613 CHQ94P 44272252 IC50 > 1000 nM T97613 CMN1U0 44272305 Ki = 0.13 nM T97613 C0LX2R 44272316 Ki = 0.05 nM T97613 C93HVQ 44272317 Ki = 0.18 nM T97613 C0VD1G 44272320 Ki = 0.22 nM T97613 CQ01LK 44272334 Ki = 4.9 nM T97613 C6NR1W 44272335 Ki = 0.94 nM T97613 CZBX31 44272406 Ki = 3.1 nM T97613 C6LP4B 44272410 Ki = 0.96 nM T97613 C60OAS 44272422 Ki = 0.2 nM T97613 C2BW8J 44272424 Ki = 11.8 nM T97613 CUX94M 44272425 Ki = 0.6 nM T97613 CUJ30W 44272430 Ki = 4.9 nM T97613 C5SVO1 44272431 Ki = 5.1 nM T97613 CO1GB4 44272438 Ki = 1.3 nM T97613 CQ9L6O 44272440 Ki = 0.35 nM T97613 CP1OX9 44272443 Ki = 1.8 nM T97613 C0L7ME 44272444 Ki = 3.5 nM T97613 C1B9MP 44272451 IC50 > 1000 nM T97613 C4SXT1 44272486 IC50 = 116 nM T97613 CCW2B6 44272487 IC50 > 1000 nM T97613 C8GYN2 44272497 IC50 > 1000 nM T97613 CZU41O 44272520 IC50 > 1000 nM T97613 CLPA83 44272521 IC50 > 1000 nM T97613 C69SPD 44272539 IC50 > 1000 nM T97613 CO76HL 44272589 IC50 > 1000 nM T97613 C8MZP1 44272590 IC50 > 1000 nM T97613 CB82FD 44272591 IC50 = 44.5 nM T97613 CI3WK7 44309030 Ki > 1000 nM T97613 C67MUK 44309034 Ki > 1000 nM T97613 C2ID4J 44317725 Ki = 7.7 nM T97613 CQ7C3V 44317822 Ki = 8.1 nM T97613 CF8K5Q 44317845 Ki = 0.39 nM T97613 CXD7H1 44340895 IC50 = 25.12 nM T97613 CH3RO2 44347098 Ki = 489.78 nM T97613 C3TBX1 44348996 Ki = 4.5 nM T97613 CMF80O 44349100 Ki = 0.63 nM T97613 CV9M5R 44349171 Ki = 75 nM T97613 CW9I4V 44349258 Ki = 50 nM T97613 C3OJ1M 44349269 Ki = 194 nM T97613 CDJ7X9 44349270 Ki = 34 nM T97613 C5DGU1 44349294 Ki = 340 nM T97613 CSA4U3 44349305 Ki = 23 nM T97613 CC92NR 44349329 Ki = 492 nM T97613 CW6U7K 44349362 Ki = 44 nM T97613 CLTG60 44353165 Ki = 1.3 nM T97613 CUQE30 44357899 Ki = 67 nM T97613 CYT31X 44358035 Ki = 49.4 nM T97613 CEB6M2 44358087 Ki = 129 nM T97613 CWT62A 44358088 Ki = 202 nM T97613 C9SHE8 44358146 Ki = 0.14 nM T97613 CPE31J 44358184 Ki = 1.5 nM T97613 CR21BK 44358196 Ki = 0.18 nM T97613 C4RVX3 44358217 Ki = 21 nM T97613 CTXM75 44358218 Ki = 17.7 nM T97613 CQE7S2 44358231 Ki = 7 nM T97613 C9JGW6 44358238 Ki = 2.2 nM T97613 CGR39W 44358274 Ki = 0.9 nM T97613 CTE2X3 44358275 Ki = 6.6 nM T97613 CSY8C4 44358276 Ki = 4.4 nM T97613 C3AJU1 44358312 Ki = 6 nM T97613 CZA67N 44358743 IC50 = 50.12 nM T97613 CZU8S4 44358744 IC50 = 158.49 nM T97613 CAQJ40 44358768 IC50 = 39.81 nM T97613 C89ZCG 44358830 IC50 = 12.59 nM T97613 CIB6Z3 44358840 IC50 = 39.81 nM T97613 CG5C2W 44358869 IC50 = 1000 nM T97613 C96IYC 44358879 IC50 = 79.43 nM T97613 CWK47R 44358887 IC50 = 1258.93 nM T97613 C5W0DJ 44358896 IC50 = 316.23 nM T97613 C28RAZ 44358910 IC50 = 199.53 nM T97613 C14HMG 44358928 IC50 = 15848.93 nM T97613 C1U3RA 44358943 IC50 = 316.23 nM T97613 CQ5XS4 44358944 IC50 = 1995.26 nM T97613 CFJ80L 44358970 IC50 = 7.943 nM T97613 CP2J5I 44358971 IC50 = 15.85 nM T97613 CN5K3L 44358991 IC50 = 1.995 nM T97613 C1Y7LF 44359018 IC50 = 19.95 nM T97613 CDBO87 44359019 IC50 = 25.12 nM T97613 CXV0U3 44359020 IC50 = 39.81 nM T97613 C5CR4V 44359035 IC50 = 3.162 nM T97613 CYPN85 44359046 IC50 = 1584.89 nM T97613 C3T5CK 44359047 IC50 = 10000 nM T97613 CJR9B2 44359058 IC50 = 12589.25 nM T97613 C9BW4I 44359070 IC50 = 15848.93 nM T97613 CD7MQ8 44359079 IC50 = 125.89 nM T97613 CR49ZP 44359113 IC50 = 7.943 nM T97613 CTF04A 44359120 IC50 = 501.19 nM T97613 C5W7SJ 44359121 IC50 = 6.31 nM T97613 C1QE9Z 44359126 IC50 = 0.7943 nM T97613 CTO94F 44359127 IC50 = 0.7943 nM T97613 CE5OZ8 44359205 IC50 = 15.85 nM T97613 CQ4MG9 44359206 IC50 = 125.89 nM T97613 CK74ML 44359228 IC50 = 3162.28 nM T97613 CV1Y9D 44359266 IC50 = 79.43 nM T97613 CA9NR7 44359270 IC50 = 3.162 nM T97613 C2HM7T 44359294 IC50 = 630.96 nM T97613 C46XLI 44359308 IC50 = 3.981 nM T97613 CF50HL 44359309 IC50 = 5.012 nM T97613 CU91NW 44359374 IC50 = 1584.89 nM T97613 CS5JF4 44359375 IC50 = 100000 nM T97613 C6V7XU 44359381 IC50 = 630.96 nM T97613 C5SO8J 44359390 IC50 = 12.59 nM T97613 CX8I2Q 44359427 IC50 = 12.59 nM T97613 CK12OG 44359437 Ki = 10.96 nM T97613 CEA02I 44359464 IC50 = 50.12 nM T97613 C1TLR9 44359465 IC50 = 79.43 nM T97613 CKFV12 44359466 IC50 = 100 nM T97613 C89JLS 44359479 IC50 = 25.12 nM T97613 C2O1DS 44389768 Ki = 60 nM T97613 CHS49R 44389812 Ki = 1 nM T97613 C5RTM7 44389813 Ki = 2 nM T97613 C4TYV6 44389839 Ki = 4 nM T97613 C0CD8U 44389845 Ki = 2 nM T97613 C6ZMD5 44389864 Ki = 9 nM T97613 C2LOD6 44394338 Ki = 39 nM T97613 CKY2H1 44394394 Ki = 16 nM T97613 C64MHD 44394415 Ki = 10 nM T97613 C40JFL 44394416 Ki = 23 nM T97613 CW4I0M 44394435 EC50 = 0.6 nM T97613 C2ZOS9 44394438 Ki = 2.1 nM T97613 C06JWG 44394456 Ki = 21 nM T97613 CRDH82 44394478 Ki = 105 nM T97613 CDN4K0 44394508 Ki = 11 nM T97613 CO61EF 44394532 Ki = 22 nM T97613 CY4CN6 44394535 Ki = 2.4 nM T97613 C2SKD1 44394556 Ki = 42 nM T97613 CD0XI1 44395856 IC50 > 1000 nM T97613 CRS38H 44395895 IC50 > 1000 nM T97613 C8V2YE 44395896 IC50 > 1000 nM T97613 C6CO1Q 44395915 IC50 > 1000 nM T97613 CE52QV 44396074 IC50 > 1000 nM T97613 CT8LC6 44396135 IC50 > 1000 nM T97613 CZF6N7 44396136 IC50 > 1000 nM T97613 CI2WG8 44396148 IC50 > 1000 nM T97613 CNT8E5 44396149 IC50 > 1000 nM T97613 CA9ZH4 44412063 Ki = 617 nM T97613 C7Y1FX 44412078 Ki = 2188 nM T97613 CN65SG 44412079 Ki = 1514 nM T97613 C9ZLR7 44412082 Ki = 724 nM T97613 CMD54S 44412141 Ki > 10000 nM T97613 CN9Y8X 44424017 Ki = 9.5 nM T97613 CPU57Y 44424018 Ki = 20.1 nM T97613 C2L0YH 44424019 Ki = 214.5 nM T97613 C1S7IT 44424020 Ki = 59.8 nM T97613 CJ80GI 44424021 Ki = 24.17 nM T97613 CT4C0R 44424022 Ki = 25.45 nM T97613 CHOU45 44424023 Ki = 70.1 nM T97613 C0EZV4 44424024 Ki = 83 nM T97613 C18YWB 44424025 Ki = 6470 nM T97613 C5NFQ7 44424026 Ki = 387 nM T97613 CXT3N5 44426096 Ki = 6.7 nM T97613 C0YUF3 44429441 Ki = 2.692 nM T97613 C8UYO4 44429442 Ki = 1.778 nM T97613 C7DGK2 44429443 Ki = 2.884 nM T97613 CXP8Z1 44429444 Ki = 8.71 nM T97613 CH79WZ 44429445 Ki = 15.85 nM T97613 CW7B9P 44429446 Ki = 19.5 nM T97613 CY7WU6 44429447 Ki = 3.548 nM T97613 CNDQ75 44429448 Ki = 4.169 nM T97613 CE1X8B 44429449 Ki = 10.47 nM T97613 CU2Y3J 44429450 Ki = 14.13 nM T97613 CG42LM 44429451 Ki = 33.11 nM T97613 C39FXQ 44429452 Ki = 12882.5 nM T97613 C6P4GD 44429453 Ki = 616.6 nM T97613 CQ9VS6 44429454 Ki = 954.99 nM T97613 CRY10T 44429455 Ki = 1258.93 nM T97613 C63DEA 44429456 Ki = 5888.44 nM T97613 CE49OW 44429457 Ki = 5370.32 nM T97613 CQ37OL 44436051 Ki = 7.244 nM T97613 C4DL5C 44469677 IC50 > 10000 nM T97613 C69IKT 44576399 IC50 = 189 nM T97613 CCP3T7 44576404 IC50 = 1220 nM T97613 CIQX03 44576405 IC50 > 10000 nM T97613 C74LMW 44576406 IC50 = 5320 nM T97613 C0LV5I 44579115 Ki = 82.5 nM T97613 C5VU7G 44579163 Ki = 49.8 nM T97613 C8R3KQ 44579164 Ki = 124 nM T97613 C1Y3GP 44579259 Ki = 137 nM T97613 C2R4MV 44579260 Ki = 24.7 nM T97613 CPAD41 44579261 Ki = 3830 nM T97613 CBYC81 44579296 Ki = 38.4 nM T97613 C40IDJ 44581851 Ki = 132 nM T97613 C8NO1P 44587356 Ki = 34.5 nM T97613 CB2ZQ5 44587357 Ki = 17.5 nM T97613 CR59BF 44593609 IC50 > 10000 nM T97613 C8S0ZG 44593610 IC50 = 2690 nM T97613 CD4G5Y 45267465 Ki = 1288.25 nM T97613 CV7Y5J 45268303 Ki = 11.75 nM T97613 C7LNE2 45268309 Ki = 1000 nM T97613 CV5KC1 45268310 Ki = 109.65 nM T97613 CS04YH 45268318 Ki = 5623.41 nM T97613 CDW89L 45269177 Ki = 257.04 nM T97613 CNC8W0 45269183 Ki = 257.04 nM T97613 C3UAM7 45270052 Ki = 8 nM T97613 C09LCX 46845151 Ki = 1.51 nM T97613 C3ID6J 46865422 EC50 = 9.03 nM T97613 CV97RU 46884552 Ki = 1840 nM T97613 CZ1AK8 46884553 Ki = 441 nM T97613 C2L9TZ 46884554 Ki = 8980 nM T97613 CY6X5U 46884555 Ki = 2010 nM T97613 C98CGH 46884599 Ki = 1460 nM T97613 CQAF97 46885226 Ki = 879 nM T97613 CI7Q8L 46885227 Ki = 263 nM T97613 CUF3Q1 46885228 Ki = 1172 nM T97613 CP06TV 46885286 Ki = 2930 nM T97613 CY0JL9 46885288 Ki = 2700 nM T97613 COK9Z0 46888491 EC50 = 2.38 nM T97613 C1XUG9 46888492 Ki = 0.64 nM T97613 C2EJD1 46888520 Ki = 0.79 nM T97613 CLKO39 46888521 Ki = 0.07 nM T97613 CQ51ZE 46888522 Ki = 0.37 nM T97613 C4X2NV 46935149 Ki = 109.65 nM T97613 C1ZYJ3 46935150 Ki = 0.7244 nM T97613 C13BFO 49865147 Ki = 42657.95 nM T97613 CG5X2S 49865148 Ki = 10471.29 nM T97613 CABU10 49865149 Ki = 3.631 nM T97613 C8F7NS 49865203 Ki = 48.98 nM T97613 CQW04N 49865204 Ki = 1.698 nM T97613 C71VAK 49865205 Ki = 2754.23 nM T97613 CAYG40 49865206 Ki = 5.754 nM T97613 C91NRX 49865265 Ki = 54.95 nM T97613 C5ZKD6 49865266 Ki = 2818.38 nM T97613 C8AHB3 49865267 Ki = 3630.78 nM T97613 C9NR2L 49865268 Ki = 0.9333 nM T97613 C2SM4J 49865269 Ki = 7.762 nM T97613 C8LI9V 49865270 Ki = 8.511 nM T97613 C96QKF 49865317 Ki = 120.23 nM T97613 CH9AZ5 49865318 Ki = 5.37 nM T97613 CQ08DG 49865319 Ki = 4.169 nM T97613 CNJ1M3 49865320 Ki = 81.28 nM T97613 CK6MU2 49865321 Ki = 3.09 nM T97613 C5PYK1 49865322 Ki = 9.12 nM T97613 CL4WG7 49865323 Ki = 70.79 nM T97613 CJRE71 49865324 Ki = 3.89 nM T97613 C8HN7M 49865373 Ki = 354.81 nM T97613 CTYD96 49865374 Ki = 36307.81 nM T97613 C10JEM 49865375 Ki = 346.74 nM T97613 CQ1X4S 49865376 Ki = 12022.64 nM T97613 CIET97 49865377 Ki = 11481.54 nM T97613 CA2B5F 49865378 Ki = 478.63 nM T97613 CR2E8T 49865423 Ki = 31622.78 nM T97613 C4EO5K 49865424 Ki = 74131.02 nM T97613 CDX4B0 49865425 Ki = 3715.35 nM T97613 C9LX2O 52918077 Ki = 1.4 nM T97613 CP7A1S 52918078 Ki = 3.3 nM T97613 C87COQ 52918079 Ki = 1.3 nM T97613 CJ7IF1 52918080 Ki = 9 nM T97613 C8NWT6 52953165 Ki = 52.8 nM T97613 CY5R6B 53231366 Ki = 57 nM T97613 CLNE80 53231367 Ki = 2860 nM T97613 CU79SK 53231464 Ki = 236 nM T97613 C7ZJH2 53231465 EC50 = 23.8 nM T97613 CW9OF1 53237946 Ki = 0.024 nM T97613 C58MYW 53237947 Ki = 0.013 nM T97613 CO3XJ2 53237948 Ki = 0.11 nM T97613 C7AF5C 53237949 Ki = 0.032 nM T97613 CP18VR 53237950 Ki = 1.1 nM T97613 CR9LF5 53237951 EC50 = 0.5129 nM T97613 CW9G3R 53238182 Ki = 0.88 nM T97613 C7N6RW 53238183 Ki = 0.0087 nM T97613 CU27MO 53238184 Ki = 0.0065 nM T97613 CF1OY4 53238185 Ki = 0.069 nM T97613 CB3H8J 53238186 Ki = 1.1 nM T97613 C3AG1Y 53238407 Ki = 0.057 nM T97613 CB12VT 53238408 Ki = 3 nM T97613 C2S0AN 53238409 Ki > 100 nM T97613 C67VCY 53238410 EC50 = 3.02 nM T97613 C0B2SG 53238411 Ki = 1.4 nM T97613 C12UVM 53238412 Ki = 1.3 nM T97613 C5KW2F 53310838 Ki = 20 nM T97613 C92HTZ 53310839 Ki = 0.083 nM T97613 CCA16D 53310840 Ki = 0.044 nM T97613 C53MGN 53310841 Ki = 0.026 nM T97613 CM9A6H 53310987 Ki = 0.31 nM T97613 CT7HJ5 53827707 IC50 = 2.3 nM T97613 C5Q4SP 54581170 Ki = 16 nM T97613 CC8U1V 54582194 Ki = 510 nM T97613 C0W8TR 54582195 Ki = 91 nM T97613 CMD87P 54583161 Ki = 9490 nM T97613 C3ANK6 54583162 Ki = 8295 nM T97613 CMP96I 54584154 Ki > 10000 nM T97613 C6G3KX 54584155 Ki = 10460 nM T97613 C0X1MI 54586060 Ki > 10000 nM T97613 C6MWF0 54586061 Ki = 1210 nM T97613 CO03ZV 54770909 Ki > 10000 nM T97613 C7KP3U 56653119 Ki = 0.15 nM T97613 C2RLP3 56653120 Ki = 3.9 nM T97613 CYL23N 56653479 Ki = 7.9 nM T97613 C2AVC9 56659223 Ki = 0.04 nM T97613 CH1IR9 56661499 Ki = 20.42 nM T97613 CV2RN0 56661512 Ki = 42.66 nM T97613 CG7H2A 56662798 Ki = 380.19 nM T97613 C5WP1S 56662799 Ki = 288.4 nM T97613 CCQ27N 56664925 Ki = 3.388 nM T97613 CXGW49 56671856 Ki = 19.95 nM T97613 C6OCQ1 56671857 Ki = 14.45 nM T97613 CZ56WJ 56671858 Ki = 741.31 nM T97613 C17XRI 56678563 Ki = 57.54 nM T97613 CJU8R5 56681902 Ki = 3.981 nM T97613 CDW2N1 71508232 EC50 = 8.38 nM T97613 CGS73W 71508233 EC50 = 16.3 nM T97613 CWO72Z 71508235 EC50 = 2.94 nM T97613 CP3Q5Z 71533430 Ki = 0.04 nM T97613 C6ZE5N 71540275 Ki = 19 nM T97613 C92WJY 71540389 Ki = 0.1 nM T97613 C0NZ2T 71540390 Ki = 87 nM T97613 CWH6T3 72548703 IC50 = 0.17 nM T97613 CM76EA 76313971 Ki = 32 nM T97613 CMD3V9 76317510 Ki = 71 nM T97613 CR75IF 76317511 Ki = 49 nM T97613 CJ15LR 76319554 Ki = 888 nM T97613 CS1ZW2 76332093 Ki = 256 nM T97613 CF23TN 79374977 Ki > 10000 nM T97613 C6KAF4 81689735 Ki = 709 nM T97613 C3M7TG 85880795 Ki = 1.2 nM T97613 CG0V6I 86272984 Ki > 1000 nM T97613 C3GYF8 86272986 Ki > 1000 nM T97613 C82OPI 86272988 Ki > 1000 nM T97613 CHK4C2 86272990 Ki > 1000 nM T97613 CU78IJ 86273221 Ki > 1000 nM T97613 C2EK6O 86273222 Ki = 170 nM T97613 CBL0V9 86273223 Ki = 280 nM T97613 CSC62G 86273226 Ki = 5 nM T97613 CDG2J4 86273227 Ki = 14 nM T97613 CY4N2D 86273228 Ki = 2.5 nM T97613 CJHY29 86273229 Ki = 17 nM T97613 CT6U5G 86273470 Ki > 1000 nM T97613 CHMV24 90655902 Ki = 0.18 nM T97613 CAT42J 90666302 Ki = 251.19 nM T97613 CBF12L 90666303 Ki = 181.97 nM T97613 CHY40Z 90666304 Ki = 57.54 nM T97613 CFMG86 90666305 Ki = 281.84 nM T97613 C1W2ZM 90666306 Ki = 5.623 nM T97613 CB4TU6 90666307 Ki = 23.99 nM T97613 CM98LH 90666308 Ki = 61.66 nM T97613 CVR1U5 90666309 Ki = 112.2 nM T97613 C4FMX7 102361822 EC50 = 396500 nM T97613 CJR85X 118712349 Ki > 10000 nM T97613 CKM9T6 118712350 Ki > 10000 nM T97613 CCY6M7 118712351 Ki > 10000 nM T97613 CM40LO 118712352 Ki > 10000 nM T97613 CFK26G 118712353 Ki > 10000 nM T97613 C4QAV9 118712354 Ki > 10000 nM T97613 C5TK7E 118712355 Ki > 10000 nM T97613 C42HKY 118712356 Ki > 10000 nM T97613 CB2RV5 118712357 Ki > 10000 nM T97613 C9Q5MI 118712358 Ki > 10000 nM T97613 C7C6SW 118712359 Ki = 500 nM T97613 CVA4W3 118712360 Ki > 10000 nM T97613 CZ7HD5 118712361 Ki > 10000 nM T97613 C1INH7 118712362 Ki > 10000 nM T97613 CWV7N2 118712363 Ki > 10000 nM T97613 C8V6WQ 118712364 Ki > 10000 nM T97613 CH9BF2 118712365 Ki > 10000 nM T97613 CKG94Y 118712366 Ki > 10000 nM T97613 CR51PL 118712367 Ki > 10000 nM T97613 CTQ8O1 118712368 Ki > 10000 nM T97613 C2G3AN 118712369 Ki > 10000 nM T97613 CGF6R8 118712370 Ki > 10000 nM T97613 CKF3O6 118712371 Ki > 10000 nM T97613 C0X1MH 118712372 Ki = 670 nM T97613 C8EJ3U 121231413 Ki = 17 nM T97613 C9AOZ2 122178507 Ki = 210 nM T97613 C7YDM4 122178508 Ki = 570 nM T97613 CZMA87 122178509 Ki = 35 nM T97613 C60SIG 122178510 Ki > 1000 nM T97613 CNI19Q 122178511 Ki > 1000 nM T97613 C1NI7Q 122178512 Ki > 1000 nM T97613 C73KSA 122178513 Ki > 1000 nM T97613 C65MIF 122188224 Ki = 57 nM T97613 C1D5YG 122188225 Ki = 13 nM T97613 CQDA72 122188226 Ki = 480 nM T97613 C07NOI 122188227 Ki = 115 nM T97613 C2H9BW 122188228 Ki > 1000 nM T97613 CYM97B 122188229 Ki = 305 nM T97613 C9D4EG 122188230 Ki = 5 nM T97613 C2XDZ5 122188231 Ki = 5.3 nM T97613 C39BDA 122188232 Ki = 132 nM T97613 CQ2OE6 122188233 Ki = 186 nM T97613 C0B2CF 122188234 Ki = 214 nM T97613 COL0N6 122188235 EC50 = 36 nM T97613 CBHP82 122188236 EC50 = 31 nM T97613 CCWU43 122188237 Ki = 45 nM T97613 CEO82Y 122188238 Ki = 122 nM T97613 C0T5HC 122188239 Ki = 291 nM T97613 CQ2IM5 122188345 Ki = 633 nM T97613 C87HOG 122188346 Ki = 0.03 nM T97613 CT1W9K 122188347 Ki = 0.7 nM T97613 CVWI64 122188348 Ki = 171 nM T97613 CT8Q6L 122188349 EC50 = 2 nM T97613 CH20AM 122188350 Ki > 10000 nM T97613 C7ND2O 122188351 Ki = 1.6 nM T97613 CBHY85 122188352 Ki = 22 nM T97613 CH3M0G 122188353 Ki = 326 nM T97613 C3JO1V 122188354 Ki > 10000 nM T97613 CPT16O 122193492 Ki = 13 nM T97613 CV5L0S 122220128 Ki = 1.905 nM T97613 CWV9T8 127025170 Ki = 210 nM T97613 CU67PG 127025781 Ki = 73 nM T97613 C0SAG6 127025782 EC50 = 8.1 nM T97613 CG53JK 127025783 Ki = 9.9 nM T97613 C7P8JY 127025784 Ki = 5.7 nM T97613 CK92ZA 127025786 EC50 = 75 nM T97613 C3YG1L 127025787 Ki = 17 nM T97613 C56JXR 127025788 Ki = 43 nM T97613 CL24NY 127026062 Ki = 2.1 nM T97613 CC87HM 127026423 Ki = 2.8 nM T97613 C7Z0HG 127026424 Ki = 10 nM T97613 CBHW31 127026425 EC50 = 1 nM T97613 C4CFA1 127026426 EC50 = 5.2 nM T97613 CQ85ZK 127026427 EC50 = 1 nM T97613 C3EA0C 127027022 Ki = 140 nM T97613 CB8RL9 127029516 Ki = 4.6 nM T97613 C4C7RU 127038129 Ki = 5 nM T97613 CY2JR9 127038130 Ki = 9 nM T97613 CU1KI9 127038131 Ki = 35 nM T97613 CO45XY 127038132 Ki = 9 nM T97613 CV0C2N 127038225 Ki = 120 nM T97613 CDV69R 127039212 Ki = 198 nM T97613 C2HQC8 127039218 Ki = 73 nM T97613 CYKA08 127040021 Ki = 2.2 nM T97613 C90XDV 127040022 Ki = 31 nM T97613 CPC79R 127040355 Ki = 68 nM T97613 C9RW7G 127041168 Ki = 6.166 nM T97613 CLK51B 127041169 Ki = 1.2 nM T97613 CYKA14 127041170 Ki = 11.75 nM T97613 CW73LQ 127042142 Ki = 0.04 nM T97613 CS0H8W 127042442 Ki = 0.2 nM T97613 COC3L8 127042791 Ki = 0.2 nM T97613 CFS87E 130400672 Ki = 430 nM T97613 CF1EZ3 137631636 Ki = 3.4 nM T97613 CR21JG 137633839 Ki = 575 nM T97613 CW39EH 137636079 Ki = 20 nM T97613 C6F1NM 137636173 Ki = 19 nM T97613 C7RUG3 137636213 Ki = 0.8 nM T97613 CX1OZ0 137637541 Ki = 62 nM T97613 CK0QM8 137637884 EC50 = 20 nM T97613 CT6EV9 137639112 Ki = 2 nM T97613 CV5QE0 137640407 Ki = 34 nM T97613 C6FPB9 137640743 Ki = 58 nM T97613 CK4I2U 137641357 Ki = 1.58 nM T97613 C0S6VY 137642160 Ki = 5 nM T97613 CUT89N 137644121 Ki = 28 nM T97613 C4Y3XB 137645530 Ki = 7 nM T97613 CAF5K6 137645887 Ki = 59 nM T97613 CEQG70 137646628 Ki > 10000 nM T97613 C3U5GH 137647756 Ki = 0.6 nM T97613 CRS5I9 137648419 Ki = 3.5 nM T97613 CL8W1O 137650611 Ki = 8 nM T97613 C19KPO 137650826 Ki = 4 nM T97613 CQDC47 137653199 Ki = 83 nM T97613 C5ST3G 137655126 Ki > 10000 nM T97613 CRF49O 137655238 Ki = 2 nM T97613 CN51KY 137655435 Ki = 60 nM T97613 CH4EL7 137655489 Ki = 315 nM T97613 CU74BT 137656715 Ki = 246 nM T97613 CQZ1T6 137656978 Ki = 892 nM T97613 COG2K4 137657824 Ki = 690 nM T97613 CZFQ41 137660180 Ki = 124 nM T97613 C5TEM2 137660333 Ki = 0.3 nM T97613 CJE60O 137660726 Ki = 16 nM T97613 CDV21J 137661786 Ki = 29 nM T97613 CAP26G 139030523 EC50 = 320 nM T97613 COD7T0 145963877 Ki = 21.38 nM T97613 COZ43N 145964105 Ki = 12.88 nM T97613 CF0BH4 145965883 Ki = 446.68 nM T97613 CSN71J 145966403 Ki = 34.67 nM T97613 CUM9C5 145966622 Ki = 0.7762 nM T97613 C5U7FM 145968467 Ki = 58.88 nM T97613 C2VK6W 145969866 Ki = 38.9 nM T97613 C26RKN 145971624 Ki = 16.22 nM T97613 CH7PT9 145971692 Ki = 370 nM T97613 C0N8ZF 145972981 Ki = 6.026 nM T97613 C6VB5Z 145974583 Ki = 3090.3 nM T97613 CZC60H 145975938 Ki = 29.51 nM T97613 CQ2Z7C 145976009 Ki = 4.898 nM T97613 C5YP8W 145976375 Ki = 27.54 nM T97613 CQAB74 145977894 Ki = 186.21 nM T97613 CC95GZ 145978811 Ki = 31.62 nM T97613 C6RV3M 145979282 Ki = 3 nM T97613 CUM97N 145979585 EC50 = 0.9 nM T97613 CV8K7E 145979689 Ki = 1 nM T97613 CM7D2G 145981162 Ki = 0.3 nM T97613 C1YJ0P 145981769 EC50 = 0.05 nM T97613 CH5A3J 145982070 Ki = 0.1 nM T97613 C9R8FK 145982167 Ki = 0.8 nM T97613 C6I5AL 145982333 Ki = 0.4 nM T97613 CO7R2A 145983175 Ki = 29 nM T97613 CF8T9A 145983929 Ki = 5 nM T97613 CM2C9Z 145986330 Ki = 6 nM T97613 C7VJ9I 145986532 Ki = 0.3 nM T97613 C3D6RX 145986700 Ki = 4 nM T97613 C7U2SG 145987794 Ki = 2 nM T97613 C7C6XZ 145988269 Ki = 2 nM T97613 CC83DQ 145988741 Ki = 0.6 nM T97613 C5Q8HG 145988801 Ki = 4 nM T97613 CH04CY 145990308 EC50 = 20 nM T97613 CRH4A6 145990662 Ki = 0.8 nM T97613 C2NF4G 145991111 Ki = 7 nM T97613 C73PGR 145991966 Ki = 2 nM T97613 CU94SI 145992795 Ki = 9 nM T97613 CX8HD4 145993188 Ki = 0.6 nM T97613 CZLY96 145993214 EC50 = 0.2 nM T97613 C43VNT 145993566 Ki = 5 nM T97613 D00RNZ 910172 Ki = 445 nM T97613 D01LAU 4284525 IC50 = 1000 nM T97613 D01SNS 4172142 Ki = 4.47 nM T97613 D01UIY 46885284 Ki = 183 nM T97613 D03AJW 44349108 Ki = 9.9 nM T97613 D03NND 22718564 Ki = 6.6 nM T97613 D03OGA 71533431 Ki = 0.03 nM T97613 D04BLO 57381112 Ki = 0.0537 nM T97613 D04VGL 3976006 Ki = 59 nM T97613 D05EDR 11630146 Ki = 1.67 nM T97613 D05TRX 22718561 Ki = 9 nM T97613 D05WKI 10244841 Ki = 1.349 nM T97613 D05ZUX 44207909 Ki >= 1000 nM T97613 D06AUM 9806449 Ki = 0.6 nM T97613 D07BKH 9798456 Ki = 275 nM T97613 D07EOD 22133318 Ki = 82 nM T97613 D07MFG 9957516 Ki = 0.55 nM T97613 D07YFL 24954989 EC50 = 0.021 nM T97613 D07ZQU 46884598 Ki = 257 nM T97613 D08SGV 10849065 Ki = 16.98 nM T97613 D08TBF 71508234 Ki = 39.5 nM T97613 D09ETU 46885285 Ki = 400 nM T97613 D09LPG 44208891 Ki = 90.4 nM T97613 D0B8PD 1858 Ki = 11.4 nM T97613 D0C5XQ 1832 Ki = 210 nM T97613 D0D6IK 10104923 Ki = 85.4 nM T97613 D0F6CD 5202 Ki > 100000 nM T97613 D0F6VI 46885230 Ki = 379 nM T97613 D0H6YF 115348 Ki = 0.013 nM T97613 D0I4DJ 24763223 Ki = 1.17 nM T97613 D0K1HD 24750192 Ki = 0.8128 nM T97613 D0L9YA 22718532 Ki = 30 nM T97613 D0O2GK 10059864 Ki = 0.15 nM T97613 D0OY8Y 11185529 Ki = 6.166 nM T97613 D0Q0LH 9998187 Ki = 27 nM T97613 D0Q6HT 11536239 Ki = 1.12 nM T97613 D0R5JD 9870523 Ki = 0.5 nM T97613 D0RF4L 129776 Ki = 32.7 nM T97613 D0S3NS 25210130 Ki = 101 nM T97613 D0S6SN 1864 Ki = 40.2 nM T97613 D0T2RY 9948320 Ki >= 1000 nM T97613 D0TM0N 24749950 Ki = 776.25 nM T97613 D0U8OS 10750842 Ki = 23.3 nM T97613 D0V7VF 16094584 Ki = 2.692 nM T97613 D0W7ZB 46885283 Ki = 1280 nM T97613 D0WE4C 5311198 Ki = 66 nM T97613 D0Y2JY 53238181 EC50 = 4.467 nM T55068 D0S6QR 214350 EC50 = 2400 nM T55068 D0X7GL 121892 EC50 = 800 nM T55068 C30IVC 155491024 EC50 = 1070 nM T55068 CTJ34I 155491025 EC50 = 350 nM T55068 C6R4FC 155513238 EC50 = 1370 nM T55068 C12LAI 155521071 EC50 = 2430 nM T55068 C8T4QV 155567226 EC50 = 1680 nM T75890 D09QOR 43157 IC50 = 14 nM T75890 CD60EW 78145 IC50 = 200 nM T75890 CBA7D6 99305 IC50 = 89 nM T75890 CPR2E6 99314 IC50 = 97 nM T75890 C9VJK8 15673476 IC50 = 43 nM T75890 D08EZR 69672 IC50 = 220 nM T67894 C9SYZ3 3708153 EC50 = 22300 nM T67894 C8PDE1 14686324 EC50 = 42500 nM T67894 C45BQH 132585194 EC50 = 4800 nM T11388 D0V3YT 10324367 IC50 = 40 nM T11388 D0X9CH 3010818 IC50 = 630 nM T11388 D07BIK 25102841 IC50 = 34.5 nM T11388 D08CJK 1150 IC50 = 15000 nM T11388 D0J6AU 10152654 Ki = 0.18 nM T11388 D0HM5J 118253852 IC50 > 20000 nM T11388 D01LNG 10201696 IC50 = 0.6 nM T11388 D0T5PH 6918602 Ki = 0.041 nM T11388 CRS0U8 1327 Ki = 22 nM T11388 C0V9XB 1339 Ki = 0.7 nM T11388 C2CM3E 1717 Ki = 3.5 nM T11388 CU27VZ 12050 IC50 > 100000 nM T11388 CAX1O8 73364 IC50 = 0.11 nM T11388 CTSD41 224665 IC50 = 80000 nM T11388 C6CP3Z 419705 IC50 > 30000 nM T11388 CW61BP 444626 Ki = 80 nM T11388 C3YF4P 462382 Ki = 1.4 nM T11388 C3SQ0W 544773 IC50 = 1300 nM T11388 CD1SC3 619687 IC50 > 30000 nM T11388 C43VCT 650125 IC50 > 30000 nM T11388 CLX45E 658024 IC50 > 30000 nM T11388 C2PGW3 659486 IC50 > 30000 nM T11388 CO30BL 664118 IC50 = 3400 nM T11388 CTI60D 714958 IC50 = 400 nM T11388 C1NSU6 847357 IC50 > 30000 nM T11388 CZC0Q2 886240 IC50 > 30000 nM T11388 COYG56 914535 IC50 = 200 nM T11388 C65UJT 980235 IC50 = 6120 nM T11388 C47TIV 997317 IC50 > 30000 nM T11388 C8WM6V 997348 IC50 = 19300 nM T11388 C5LZB9 1212080 IC50 > 30000 nM T11388 C25SXA 1440071 IC50 = 3830 nM T11388 C9S6OE 1500321 IC50 = 2500 nM T11388 CZ4KG8 1584145 IC50 > 30000 nM T11388 C7G2MP 1903670 IC50 = 4300 nM T11388 CA4K6U 2443028 IC50 > 30000 nM T11388 CFB6Y7 2738067 IC50 = 13300 nM T11388 CA3K9L 2822094 IC50 = 21300 nM T11388 CZ9HF4 2822538 IC50 = 2000 nM T11388 CG9A3S 2822542 IC50 > 10000 nM T11388 C8UC6T 3128115 IC50 > 30000 nM T11388 C6NXZ0 4247255 IC50 = 5800 nM T11388 CX2ZL3 4529335 IC50 > 30000 nM T11388 CZ7W8T 5001827 IC50 > 30000 nM T11388 CJN1R6 5286932 IC50 = 21400 nM T11388 CR2ND4 5287468 Ki = 0.16 nM T11388 CW6D7Z 5287498 IC50 = 0.1288 nM T11388 CB6H0T 5287549 Ki = 0.0048 nM T11388 CESY50 5288259 IC50 = 0.83 nM T11388 C6YF4B 5288616 IC50 = 6 nM T11388 CFM6E4 5288618 IC50 = 7 nM T11388 CBNO34 5288632 Ki = 27 nM T11388 C9E1UW 5288633 Ki = 10 nM T11388 C5HE7U 5288634 Ki = 0.7 nM T11388 CN3RY0 5289345 Ki = 22 nM T11388 C6UYA0 5406325 IC50 > 30000 nM T11388 COU80Q 5704072 IC50 = 100 nM T11388 CMJA72 5723164 IC50 > 30000 nM T11388 C1CVF6 5935636 IC50 = 10500 nM T11388 C6PJ9O 5935645 IC50 > 30000 nM T11388 CI2GZ5 5941217 IC50 > 30000 nM T11388 CC84QY 5963786 IC50 > 30000 nM T11388 CH0TP8 6148373 IC50 = 1600 nM T11388 C4ZI1O 6314543 IC50 > 30000 nM T11388 C1DAZ6 6420159 Ki > 30000 nM T11388 CZEG39 6449829 IC50 = 170 nM T11388 C6XNU5 6917569 IC50 = 160 nM T11388 C0XQP7 6917747 IC50 > 100000 nM T11388 C2C5DW 6998013 IC50 = 110 nM T11388 CZIB15 7015728 IC50 = 200 nM T11388 CE6QZ8 7404011 IC50 = 5300 nM T11388 CGLR90 7431055 IC50 = 2700 nM T11388 CN26IL 9547980 Ki > 100000 nM T11388 C9GW5K 9567107 IC50 > 30000 nM T11388 CH7D8I 9609685 IC50 = 7600 nM T11388 CU1YI6 9694136 IC50 = 5800 nM T11388 CB32AH 9812750 IC50 = 100 nM T11388 C4UE3W 9813935 IC50 = 12100 nM T11388 CQ1NG7 9815041 IC50 = 56 nM T11388 CIX3A6 9816412 IC50 = 81 nM T11388 C9F7PL 9825191 Ki = 607 nM T11388 C2AI0Z 9834360 IC50 = 370 nM T11388 CLND75 9835685 IC50 = 290 nM T11388 C6R0JY 9843767 IC50 = 14000 nM T11388 CLQ92U 9848147 IC50 = 190 nM T11388 C2VX4Z 9848148 Ki = 1.8 nM T11388 C8TL5X 9855884 IC50 = 70 nM T11388 CYMA06 9856358 IC50 = 26000 nM T11388 CVS7N2 9877581 IC50 = 40 nM T11388 CC3X2P 9877623 IC50 = 20 nM T11388 CO0PD1 9883178 IC50 < 3 nM T11388 CGA91J 9890145 IC50 = 69 nM T11388 C8P5LN 9891030 Ki = 0.8 nM T11388 C5L4YE 9893225 IC50 = 40.5 nM T11388 COK50T 9895628 IC50 < 1 nM T11388 CIBS75 9899272 IC50 = 100 nM T11388 CLF3Z2 9901081 IC50 = 330 nM T11388 CW5Y9P 9901142 IC50 = 30 nM T11388 C5XS2F 9904539 Ki = 4100 nM T11388 CALH63 9908450 IC50 = 7.8 nM T11388 CA7U5T 9909950 IC50 = 230 nM T11388 CHU41G 9913263 IC50 = 3.9 nM T11388 C7WKG9 9913437 IC50 = 54 nM T11388 C78CYD 9920989 IC50 = 13700 nM T11388 CLY9Q7 9925805 IC50 = 16 nM T11388 CT74FA 9933804 IC50 = 0.5 nM T11388 C5ZD9R 9943969 IC50 = 6 nM T11388 CNR6D5 9948720 IC50 = 1030 nM T11388 C0PJ2U 9964915 IC50 = 17 nM T11388 CLMJ35 9967252 IC50 = 480 nM T11388 C4WFJ2 9980678 Ki = 25 nM T11388 CBNR45 9980918 IC50 = 6.4 nM T11388 CHN80D 9981917 IC50 < 3 nM T11388 CT2A7L 9983757 Ki = 790 nM T11388 C1F4BA 9984481 IC50 = 840 nM T11388 C1ZUE0 9999103 Ki = 14 nM T11388 CGM73V 10000717 Ki = 19 nM T11388 CQ0J8M 10003594 IC50 = 3 nM T11388 C7P6JO 10004326 IC50 < 1 nM T11388 C40APB 10005577 IC50 = 3.6 nM T11388 CI96RJ 10008050 IC50 = 136 nM T11388 CXY9N8 10024008 IC50 = 7.3 nM T11388 CLB5G0 10025017 IC50 = 3 nM T11388 C4NW7I 10026902 IC50 = 3.7 nM T11388 CF95YG 10027990 IC50 = 1.6 nM T11388 CT26WE 10030928 Ki = 0.8 nM T11388 C0SJY5 10031327 IC50 = 174 nM T11388 CJO52T 10046162 IC50 < 1 nM T11388 CU1EF5 10047111 IC50 = 5 nM T11388 C68HGW 10047261 IC50 = 0.2 nM T11388 C8F7MU 10047536 IC50 = 3.8 nM T11388 CGX58K 10051123 IC50 = 1 nM T11388 CXH45E 10051341 IC50 = 1 nM T11388 CG39EA 10059139 IC50 = 52000 nM T11388 C2N9CS 10062713 IC50 = 0.5 nM T11388 C6O8RU 10072812 IC50 = 7.5 nM T11388 CV29YC 10076076 IC50 = 2300 nM T11388 CHV2M3 10077641 Ki = 1.9 nM T11388 CHA42Q 10097070 IC50 < 3 nM T11388 C9T8UM 10098687 IC50 = 3.802 nM T11388 C8FPB5 10098917 IC50 = 450 nM T11388 CSO9B2 10099774 Ki = 3.5 nM T11388 CY6Q1M 10108990 IC50 = 950 nM T11388 C57JDN 10118049 IC50 = 4.7 nM T11388 CFC3Q8 10120133 IC50 = 0.3715 nM T11388 C6AZ3B 10120903 IC50 = 5800 nM T11388 C97NJR 10121949 Ki = 550 nM T11388 C7XOA0 10127183 IC50 = 0.9 nM T11388 CSO96K 10127748 IC50 = 8.5 nM T11388 CI4V3K 10128045 IC50 = 260 nM T11388 CVPJ85 10128987 IC50 = 54 nM T11388 CKZ15P 10129236 IC50 = 13 nM T11388 C9WRK0 10129345 IC50 = 31 nM T11388 C9EG5U 10131775 IC50 = 4.2 nM T11388 CJ79ZX 10138553 IC50 = 20 nM T11388 CY6PU1 10143615 Ki = 4 nM T11388 CLID02 10144235 Ki = 29 nM T11388 CQ3YD8 10150891 IC50 = 0.2 nM T11388 C7AV3P 10152318 IC50 = 11 nM T11388 C0Y9WT 10152540 IC50 = 85 nM T11388 CN6OH8 10152709 IC50 = 1900 nM T11388 C8DQG0 10154619 IC50 = 52 nM T11388 CO2Z7G 10155296 IC50 = 3 nM T11388 C9VFI4 10161284 IC50 = 2.3 nM T11388 C1Q2EX 10164497 Ki = 7.9 nM T11388 CDX7R4 10164961 IC50 = 830 nM T11388 CY06GM 10164962 IC50 = 0.8318 nM T11388 C5B1HM 10165557 IC50 = 0.2399 nM T11388 C09ALX 10165785 Ki = 0.0099 nM T11388 CR62PT 10165786 Ki = 19 nM T11388 CXHS80 10165939 IC50 = 0.6457 nM T11388 CTJ7R3 10166544 IC50 = 0.0257 nM T11388 CDRE91 10167323 Ki = 22 nM T11388 CZ1A8U 10173731 IC50 = 0.2 nM T11388 C5NEX6 10174161 IC50 = 26 nM T11388 C1YR4T 10174359 IC50 = 16.98 nM T11388 C07GUT 10184761 Ki = 1.3 nM T11388 C4M3SG 10186046 IC50 = 4900 nM T11388 CCO7A6 10187105 Ki = 1300 nM T11388 CP2M1T 10187189 Ki = 1.5 nM T11388 C9WTI5 10187190 Ki = 42 nM T11388 C0SF7U 10187920 IC50 = 0.02512 nM T11388 C9T5PN 10190977 IC50 = 98 nM T11388 CUFY02 10193166 IC50 = 350 nM T11388 CKZ1A0 10194354 IC50 = 0.3 nM T11388 CZD7A6 10194447 IC50 = 0.3 nM T11388 CG7B9T 10194508 IC50 = 17 nM T11388 CA2UH4 10194634 IC50 = 0.6 nM T11388 C49OCV 10195734 IC50 = 37 nM T11388 CWPU45 10196366 IC50 = 98 nM T11388 C4A6PK 10196730 IC50 = 54 nM T11388 C1NCJ2 10196913 IC50 = 230 nM T11388 CO7XD6 10198366 IC50 = 10 nM T11388 C5T8PK 10198752 IC50 = 20 nM T11388 CL9DW3 10200425 IC50 = 9 nM T11388 CS3IP7 10210867 IC50 = 0.4074 nM T11388 C1WL9J 10211340 Ki = 54 nM T11388 CAH08N 10214815 IC50 = 140 nM T11388 C87PIY 10214967 IC50 = 21 nM T11388 CF2XJ7 10215685 IC50 = 150 nM T11388 CB2XL0 10215686 IC50 = 33 nM T11388 C1F9SP 10216231 IC50 = 44 nM T11388 C1Y3QZ 10216510 IC50 = 0.1 nM T11388 C5GSN6 10216511 IC50 = 0.5 nM T11388 CE6K2Q 10230391 IC50 = 460000 nM T11388 CT8K5D 10231379 IC50 = 0.072 nM T11388 C4OZ5K 10231447 IC50 = 0.02884 nM T11388 CJBI61 10237771 IC50 = 0.8 nM T11388 CFI43Z 10238903 IC50 = 0.2 nM T11388 CC8QG6 10239612 IC50 = 51 nM T11388 CZ0A1F 10241556 IC50 = 58 nM T11388 CORW86 10247897 IC50 = 3.2 nM T11388 CEQ21I 10249499 IC50 = 8.6 nM T11388 C6A8NV 10252643 Ki = 4 nM T11388 CD0QG1 10253693 IC50 = 3.8 nM T11388 CWG70R 10256998 IC50 = 6.607 nM T11388 CB32HU 10262225 IC50 = 38 nM T11388 CJ19AP 10264740 IC50 = 30 nM T11388 CEZ0A6 10269099 IC50 = 200 nM T11388 CH14BY 10269694 IC50 = 110 nM T11388 C9SOH2 10271564 IC50 = 57 nM T11388 CBHO04 10272927 IC50 < 1 nM T11388 CKX0R7 10287617 IC50 = 0.9 nM T11388 CUW38E 10288162 IC50 = 1.1 nM T11388 CX23AL 10288163 IC50 = 6 nM T11388 CY7DQ2 10288811 IC50 = 23.99 nM T11388 CJ4U7Y 10289785 IC50 = 50 nM T11388 CV9LB1 10302710 IC50 = 1500 nM T11388 CUQ2R3 10303526 IC50 = 8100 nM T11388 CV5S7B 10303657 IC50 = 5800 nM T11388 CZR02J 10303878 Ki = 37 nM T11388 CYKL86 10308326 IC50 = 990 nM T11388 CJ05UY 10308440 IC50 = 100 nM T11388 CAV8Y5 10308447 IC50 = 700 nM T11388 CO20DN 10308576 IC50 = 28 nM T11388 CZ0Y9P 10308614 IC50 = 30 nM T11388 CPT49O 10310362 IC50 = 0.4 nM T11388 CMR18K 10310975 IC50 = 210 nM T11388 C89EQT 10311492 IC50 > 12000 nM T11388 C5KBT6 10311986 IC50 = 87 nM T11388 CO0GQ8 10313520 IC50 = 360 nM T11388 CWS2D6 10316842 IC50 = 0.77 nM T11388 C9DN6G 10325113 IC50 = 44.5 nM T11388 C59ZDR 10337631 IC50 = 10 nM T11388 C2GLK6 10346121 IC50 = 6.5 nM T11388 CXMY07 10347335 IC50 = 8.318 nM T11388 CI0ET1 10348741 Ki = 0.6 nM T11388 CY60AW 10367515 IC50 = 2.7 nM T11388 CDX2C8 10367993 IC50 = 7.1 nM T11388 CYF98Z 10368089 IC50 < 3 nM T11388 CBMA02 10388992 IC50 = 410 nM T11388 CX7S8A 10392779 IC50 = 1100 nM T11388 C25DTV 10393262 IC50 = 4.8 nM T11388 CJ3TN7 10413773 IC50 = 4.5 nM T11388 C41JUO 10414118 IC50 = 9 nM T11388 CDVZ19 10431266 Ki = 5.7 nM T11388 C57DYJ 10437715 Ki = 10 nM T11388 CH4LQ2 10437784 IC50 = 6.4 nM T11388 CZ3R0W 10453897 IC50 = 2.512 nM T11388 CN18SE 10456222 Ki = 0.74 nM T11388 C06QJW 10457653 IC50 = 8.4 nM T11388 C8G9SX 10458632 IC50 = 5.6 nM T11388 CK9PX5 10461097 Ki = 0.5 nM T11388 C5M7BL 10471316 IC50 = 8.6 nM T11388 CXD68E 10473874 IC50 = 7.2 nM T11388 C42PHV 10474557 Ki = 15 nM T11388 C9D7XO 10478741 IC50 = 1.7 nM T11388 C32MAD 10482525 IC50 = 28.2 nM T11388 C9M2RV 10483128 Ki = 1.4 nM T11388 COVN15 10484214 Ki = 33 nM T11388 C1MX2S 10499322 Ki = 44 nM T11388 C2S8XD 10506997 Ki = 3.4 nM T11388 CHTL13 10507714 Ki = 2 nM T11388 CZ80TL 10507960 Ki = 8200 nM T11388 CGA7D1 10515827 IC50 = 200 nM T11388 C25HQJ 10522795 Ki > 1000 nM T11388 C0UBF5 10524384 Ki = 250 nM T11388 CZUA37 10531571 Ki = 3500 nM T11388 C5HB0R 10553858 Ki = 670 nM T11388 CR54HQ 10569603 Ki > 10000 nM T11388 C8U1RQ 10593841 Ki = 140 nM T11388 C1C6UK 10604848 Ki = 54 nM T11388 CLUJ05 10627524 Ki = 56 nM T11388 CM61OV 10627712 Ki = 16000 nM T11388 CH38ZO 10650265 Ki = 100 nM T11388 CJTH67 10668881 Ki = 230 nM T11388 C9V5EX 10673009 Ki = 7.5 nM T11388 C5BUY2 10674052 Ki = 1 nM T11388 CRL23A 10674588 Ki = 1.4 nM T11388 C6GX2C 10676280 Ki = 4.7 nM T11388 C9PY4N 10690022 Ki = 150 nM T11388 CKO6L0 10698950 Ki = 2.6 nM T11388 CB54AK 10717998 Ki = 120 nM T11388 CDS3M7 10722309 Ki = 1.6 nM T11388 C67NAM 10746468 Ki = 15000 nM T11388 CXB2Y7 10768964 Ki = 12 nM T11388 CP42MK 10792226 Ki = 0.16 nM T11388 C3TXU5 10792279 Ki > 1000 nM T11388 C9AIY1 10793962 Ki = 180 nM T11388 CQ08YK 10807774 Ki > 1000 nM T11388 CHC3F0 10817683 Ki = 15 nM T11388 CZ4V0F 10832380 Ki > 10000 nM T11388 C78VEK 10837067 Ki = 25 nM T11388 CJO1U8 10848617 IC50 = 36 nM T11388 CBWJ85 10862359 IC50 = 6 nM T11388 CNVG58 10875013 IC50 < 3 nM T11388 CPAF53 10876251 Ki = 6.76 nM T11388 C7YTP5 10887117 Ki = 2.12 nM T11388 CZK49P 10893343 IC50 = 291 nM T11388 CTZ4G0 10898089 Ki = 8.42 nM T11388 C6WUK7 10898110 Ki = 2.45 nM T11388 CWXN58 10902758 Ki > 100000 nM T11388 CBJ1I7 10902914 IC50 = 1036 nM T11388 CA30HS 10905508 IC50 = 65 nM T11388 CV0Z7C 10906068 IC50 < 3 nM T11388 CIFW32 10916659 IC50 > 1000 nM T11388 C5X6NA 10924832 IC50 = 488 nM T11388 C2CYZ8 10927418 IC50 = 460 nM T11388 C3VN9H 10931029 Ki = 100 nM T11388 CTJG76 10938642 IC50 > 1000 nM T11388 CZG37Y 10938664 IC50 = 51 nM T11388 CDE53Q 10960298 IC50 = 190 nM T11388 CL7W4P 10960628 IC50 = 14 nM T11388 CW1L5K 10960899 IC50 < 3 nM T11388 CR0P8J 10971179 IC50 = 87 nM T11388 CK9E8W 10972182 IC50 = 1405 nM T11388 C6ZOI1 10979734 IC50 = 803 nM T11388 C57TZJ 10985562 Ki = 0.86 nM T11388 CA3NG9 10993428 IC50 = 62 nM T11388 C4E0HT 11007209 Ki = 0.18 nM T11388 CM9Z5T 11012257 IC50 = 142 nM T11388 C5UMF7 11013396 IC50 = 79 nM T11388 C5XHI0 11014664 IC50 = 638 nM T11388 CC6OQ2 11017520 Ki = 34 nM T11388 C2C5VH 11025400 IC50 = 470 nM T11388 CY72BF 11034349 IC50 = 1463 nM T11388 CDO18Y 11053055 IC50 = 250 nM T11388 C5C8TK 11061638 Ki = 2.13 nM T11388 C8RU9F 11067956 IC50 = 8 nM T11388 C0PSR8 11081485 IC50 = 922 nM T11388 C5WY1H 11082075 IC50 < 3 nM T11388 CQ4L0T 11122768 IC50 < 3 nM T11388 CQK6U4 11144121 IC50 = 60 nM T11388 C27OHY 11155113 IC50 = 71 nM T11388 CDR7A6 11155973 Ki = 286 nM T11388 C8EAL0 11156785 Ki = 995 nM T11388 C9SN1Q 11157631 Ki = 260 nM T11388 CH41OF 11157632 Ki = 5410 nM T11388 C8ZRG0 11157920 IC50 = 9 nM T11388 CK78BZ 11163617 IC50 = 12000 nM T11388 CAX52F 11164895 IC50 = 0.71 nM T11388 CM09XA 11165672 IC50 = 54 nM T11388 C61AIQ 11168385 Ki = 291 nM T11388 CAI94Q 11168613 Ki = 184 nM T11388 CXJL01 11176831 IC50 = 18 nM T11388 C2VJG7 11178623 Ki = 4560 nM T11388 CMDU74 11180007 Ki = 11530 nM T11388 COP23L 11181707 IC50 = 159 nM T11388 C41LHB 11188458 IC50 = 36 nM T11388 CUF86R 11188663 IC50 = 24 nM T11388 CO64CZ 11189948 IC50 = 0.65 nM T11388 C47XVC 11190260 IC50 = 65 nM T11388 C9ZNL4 11191320 Ki = 10.1 nM T11388 CS90MB 11191512 Ki = 217 nM T11388 CIC65O 11192788 IC50 = 9.5 nM T11388 C72VIY 11192835 IC50 = 1.6 nM T11388 CKD73X 11193068 IC50 = 2.9 nM T11388 CW50QF 11196731 IC50 = 38 nM T11388 CUN2A1 11199770 IC50 = 95 nM T11388 CT8VQ9 11200473 IC50 = 71 nM T11388 C2H4GP 11200735 Ki = 80 nM T11388 CB60IH 11201021 IC50 = 39 nM T11388 COIM61 11201464 IC50 = 1.7 nM T11388 CTCX89 11203484 Ki > 30000 nM T11388 C17UIX 11203679 IC50 = 26 nM T11388 C7ZP2Q 11204834 IC50 = 10 nM T11388 CH3Y0R 11211199 IC50 = 0.41 nM T11388 CJVI81 11214912 IC50 > 12000 nM T11388 CO5DJ2 11214953 IC50 = 0.3 nM T11388 CP0JO9 11222736 IC50 = 0.47 nM T11388 C7SOL0 11224927 Ki > 20000 nM T11388 CM8ZV1 11225780 Ki = 24290 nM T11388 CLC2X1 11226457 Ki > 100000 nM T11388 CQX39V 11233954 IC50 = 5.1 nM T11388 CA25SW 11235163 IC50 >= 12000 nM T11388 C4VFD2 11235460 IC50 = 51 nM T11388 C0JO5R 11238059 Ki > 100000 nM T11388 C3T1LM 11238468 Ki > 100000 nM T11388 CAXO42 11246702 IC50 = 68 nM T11388 C5VY1E 11247716 Ki > 30000 nM T11388 C25FSN 11247725 IC50 = 15 nM T11388 CLA6J3 11249688 Ki > 10000 nM T11388 CRXU26 11250282 Ki > 30000 nM T11388 CU05SV 11250788 IC50 = 16 nM T11388 CX8NC1 11256746 IC50 = 360 nM T11388 C67KJR 11257892 IC50 = 120 nM T11388 CHK9N2 11261516 Ki > 30000 nM T11388 C2U5ZS 11261768 IC50 = 4.2 nM T11388 CN87GA 11262606 IC50 = 6.9 nM T11388 C1T8AC 11262663 IC50 = 2.6 nM T11388 CTMQ46 11268566 IC50 = 20 nM T11388 CE12NZ 11269005 IC50 = 32 nM T11388 CTYS25 11269348 IC50 = 0.91 nM T11388 CK8MP7 11269375 IC50 = 135 nM T11388 C8F2ZN 11269453 IC50 < 1 nM T11388 CU6M9Z 11270375 IC50 = 27 nM T11388 CIFQ06 11273375 Ki = 2150 nM T11388 CM6V4X 11280517 IC50 = 47 nM T11388 C15XUE 11283547 Ki = 11530 nM T11388 CCH6N4 11283555 IC50 = 0.3 nM T11388 CM86BP 11294094 Ki > 20000 nM T11388 CFU50G 11294227 Ki > 10000 nM T11388 CV86IB 11295906 Ki > 100000 nM T11388 CI7OP4 11303107 IC50 = 350 nM T11388 CQ0ON8 11303478 IC50 = 52 nM T11388 C0AWT6 11305090 IC50 = 20 nM T11388 CZX89I 11305296 Ki > 30000 nM T11388 CR2T5B 11305867 Ki = 9340 nM T11388 CU6Z0F 11306593 Ki > 30000 nM T11388 C06JLW 11307085 IC50 = 0.2 nM T11388 CKS3Z7 11307651 IC50 = 57 nM T11388 CON02M 11314186 IC50 = 25 nM T11388 CB2GN4 11314758 IC50 = 36 nM T11388 CI0CZ5 11314946 IC50 = 1.8 nM T11388 CWE0Y1 11315122 IC50 = 83 nM T11388 CEC0A2 11316876 Ki > 30000 nM T11388 C8HIC6 11319255 IC50 = 7.3 nM T11388 C42FVC 11326873 IC50 = 26 nM T11388 CDYL91 11327594 Ki > 100000 nM T11388 CP5MI6 11329727 Ki = 3706 nM T11388 CEZ4A1 11330658 IC50 = 150 nM T11388 CET6U2 11338550 IC50 = 0.46 nM T11388 CD70PA 11341599 Ki = 1050 nM T11388 CRB7E8 11342699 IC50 = 54 nM T11388 CFO1P2 11351230 IC50 = 0.21 nM T11388 C5X1VW 11351327 IC50 = 2003 nM T11388 CFJ70U 11353015 Ki > 100000 nM T11388 C4K8FU 11354336 IC50 = 7.3 nM T11388 CY9P2B 11362165 IC50 = 15 nM T11388 CZ02MR 11362698 IC50 = 63 nM T11388 CNZ72W 11362838 IC50 = 58 nM T11388 C2FJL5 11372012 IC50 = 17 nM T11388 C07BQS 11372366 IC50 = 62 nM T11388 CD9I5L 11372367 IC50 = 3.4 nM T11388 CT9BU3 11373469 IC50 = 45 nM T11388 CVC4Z6 11373861 IC50 = 83 nM T11388 CI3T7B 11374356 IC50 = 62 nM T11388 C54OEH 11375798 IC50 = 0.2 nM T11388 C9W0TB 11375856 Ki > 30000 nM T11388 C7NQX3 11375955 Ki > 26400 nM T11388 CH4I3T 11375956 IC50 = 14 nM T11388 C34DFQ 11376188 Ki > 100000 nM T11388 CAL7B2 11376611 Ki > 100000 nM T11388 C7PT9S 11377607 IC50 = 68 nM T11388 C9UR5O 11380890 IC50 = 40 nM T11388 CMR83T 11385048 IC50 = 14 nM T11388 CG73DJ 11385151 IC50 = 17 nM T11388 CZD9I3 11385218 IC50 = 25 nM T11388 CC3NS1 11385219 IC50 = 62 nM T11388 COV1F4 11387157 Ki = 10540 nM T11388 CEW0F3 11387421 Ki = 11700 nM T11388 CDM4U7 11387844 IC50 = 4.3 nM T11388 C3DQL2 11396020 Ki > 30000 nM T11388 C4QM7I 11396148 Ki > 30000 nM T11388 CER2V8 11397519 Ki > 10000 nM T11388 C4ZLU9 11397590 Ki > 100000 nM T11388 C7RFC5 11398171 Ki = 907 nM T11388 CO43YH 11399749 IC50 = 85 nM T11388 C12SDO 11406824 IC50 = 9.2 nM T11388 C90LAC 11408098 IC50 = 10 nM T11388 CI3HK2 11409407 Ki = 14700 nM T11388 CO4Y3H 11410560 Ki > 100000 nM T11388 CU4P8A 11418931 Ki = 139 nM T11388 C56SXA 11419952 Ki = 8810 nM T11388 C0F5GE 11420649 IC50 = 61 nM T11388 CGD1K4 11421700 Ki = 8710 nM T11388 CY1SE0 11422514 IC50 = 15 nM T11388 C58WQT 11430095 IC50 = 27 nM T11388 C2IJ6G 11430812 IC50 = 22 nM T11388 CILJ37 11431699 Ki = 3706 nM T11388 CM2VQ6 11431993 Ki > 30000 nM T11388 C19YRB 11432272 Ki = 1140 nM T11388 C72PFO 11432501 Ki = 3710 nM T11388 C65ASH 11432773 Ki > 100000 nM T11388 CQRB45 11433280 Ki = 1480 nM T11388 CH65FU 11436272 IC50 = 51 nM T11388 CQIP48 11439739 IC50 = 10 nM T11388 CD21WG 11441440 IC50 = 68 nM T11388 CME0C5 11443502 Ki = 3.5 nM T11388 CH9ZA7 11443990 Ki = 2130 nM T11388 CI8Z6M 11451427 IC50 = 1200 nM T11388 C1I6LU 11452160 IC50 = 52 nM T11388 C1AT2Z 11453155 IC50 = 555 nM T11388 C0U6JW 11453603 IC50 = 0.24 nM T11388 CL53MS 11456165 Ki > 100000 nM T11388 CME32S 11456379 Ki > 37250 nM T11388 C0O8MK 11464526 IC50 = 3.5 nM T11388 C0VB9G 11464589 IC50 = 140 nM T11388 C5N3BV 11466327 Ki > 20000 nM T11388 CV43WB 11466677 Ki = 557 nM T11388 CM59AQ 11466845 Ki = 2480 nM T11388 CRM65O 11467250 IC50 = 33 nM T11388 CL1D2Z 11471738 IC50 = 1 nM T11388 CR7O3Z 11474385 IC50 = 32 nM T11388 CQCR56 11475863 IC50 = 250 nM T11388 C0ZK5I 11477975 Ki > 10000 nM T11388 C9U0YI 11478637 Ki = 710 nM T11388 C91OEA 11479185 IC50 = 8.3 nM T11388 C78JVD 11485907 IC50 = 40 nM T11388 CQ0GR8 11487339 IC50 = 0.26 nM T11388 CBC8U6 11490230 Ki = 4870 nM T11388 CS1H2J 11490661 IC50 = 3.9 nM T11388 C94SZC 11493500 Ki = 6300 nM T11388 CZLF20 11494632 Ki = 16000 nM T11388 CR2M4H 11494672 Ki = 28000 nM T11388 C5CL9A 11496988 Ki = 460 nM T11388 CC92RV 11501571 IC50 = 19 nM T11388 CFI8L5 11502586 IC50 = 2.5 nM T11388 CK5JM6 11503223 IC50 = 0.4 nM T11388 CY4A7V 11504785 Ki = 0.89 nM T11388 C3Q7BE 11504819 Ki = 30 nM T11388 CF20TJ 11514361 Ki > 100000 nM T11388 C23DKS 11516307 IC50 = 4 nM T11388 C87YFV 11523212 Ki = 83000 nM T11388 CW1G0N 11529814 IC50 = 370 nM T11388 CNH9B0 11530527 IC50 = 150 nM T11388 C7NO5X 11531213 IC50 = 10 nM T11388 CQ6UC2 11537070 Ki = 3300 nM T11388 C35CAW 11543897 IC50 = 490 nM T11388 CY0AV1 11544076 Ki = 2100 nM T11388 C98EQF 11545899 IC50 = 0.94 nM T11388 C65NQY 11550481 Ki = 5000 nM T11388 C28XJZ 11551007 IC50 = 52 nM T11388 CYO67B 11551502 Ki = 2100 nM T11388 CB3W8O 11565199 Ki = 1510 nM T11388 CYJ2E7 11574887 IC50 = 0.28 nM T11388 C9YNX2 11581727 Ki = 6500 nM T11388 C73VCU 11584899 Ki = 10.5 nM T11388 CJG6T3 11585276 Ki = 295 nM T11388 CRY5B8 11587214 IC50 = 410 nM T11388 CER65Q 11588182 Ki = 29000 nM T11388 C7MQB5 11597331 IC50 = 230 nM T11388 C1QO2C 11598043 IC50 = 140 nM T11388 CT8XH2 11603305 Ki > 100000 nM T11388 CM4OS2 11606272 Ki = 12 nM T11388 C7W8JG 11616689 Ki > 100000 nM T11388 CP0BX4 11617382 IC50 = 280 nM T11388 CG0E6F 11618082 IC50 = 460 nM T11388 CH21OU 11623464 Ki = 4100 nM T11388 C0C5SD 11624809 IC50 = 5 nM T11388 C9LBF3 11628054 Ki = 29 nM T11388 C3XO5G 11631355 Ki > 100000 nM T11388 C98QKS 11635243 Ki = 2.5 nM T11388 CNH8C7 11646581 Ki = 26000 nM T11388 C2XHN1 11646851 Ki > 100000 nM T11388 CILB73 11649751 Ki > 65000 nM T11388 C8NZX4 11651881 Ki = 3300 nM T11388 CPG5O8 11652408 IC50 = 100 nM T11388 C2PM1X 11652420 Ki > 100000 nM T11388 C5ZOM0 11656060 IC50 <= 0.005 nM T11388 CO76PW 11659287 Ki = 90000 nM T11388 CC6FP9 11659805 IC50 = 200 nM T11388 CG3W2T 11666681 IC50 = 8 nM T11388 CSD3H5 11666846 Ki = 8500 nM T11388 C23WER 11667717 IC50 = 2.6 nM T11388 C5SJ9K 11669355 IC50 = 100 nM T11388 CY52ZR 11670661 IC50 = 1 nM T11388 CKH3O7 11673861 Ki > 1000000 nM T11388 C23ZVP 11678241 Ki = 52 nM T11388 C27LJY 11678922 Ki > 10000 nM T11388 CL4XB1 11685284 Ki = 1.4 nM T11388 C53OYX 11692372 Ki = 0.14 nM T11388 C6F1GI 11695261 Ki = 5300 nM T11388 C5H2GL 11696621 Ki = 4200 nM T11388 C7QIP8 11699507 Ki = 4.5 nM T11388 C45DTR 11702249 Ki = 74 nM T11388 CRTS62 11703216 Ki = 34000 nM T11388 C5UEI7 11703527 IC50 = 4 nM T11388 C9X6PV 11703830 Ki = 2.2 nM T11388 CRZ6T0 11709547 Ki = 13000 nM T11388 CT4QY5 11710096 Ki = 66000 nM T11388 C5FZ1J 11710873 IC50 = 3 nM T11388 C5ME9N 11716536 Ki = 1200 nM T11388 CMQ35I 11726291 IC50 = 1.9 nM T11388 C93ZBQ 11729403 Ki = 61 nM T11388 CDS4P0 11743922 Ki = 30 nM T11388 C1KU9M 11750163 IC50 = 17 nM T11388 C76VZC 11750525 IC50 = 76 nM T11388 C0SV2T 11753412 Ki = 16700 nM T11388 C78GRH 11755837 IC50 = 17 nM T11388 CQJ98N 11756263 IC50 = 4.8 nM T11388 C1IVT2 11756512 IC50 = 4.266 nM T11388 CXZI19 11757462 IC50 = 16.98 nM T11388 CD73UO 11768265 Ki = 72 nM T11388 C8D7BS 11771234 Ki = 18000 nM T11388 CD18PM 11772556 IC50 = 1.6 nM T11388 CR2C5L 11774667 IC50 = 4.8 nM T11388 CC8K5W 11775397 IC50 = 22 nM T11388 CT5B1S 11784942 Ki > 100000 nM T11388 CV1KZ3 11799129 Ki = 1.6 nM T11388 CDJH89 11811557 IC50 = 8 nM T11388 CLY2A4 11811595 IC50 = 840 nM T11388 CQFU14 11811813 IC50 = 350 nM T11388 CZ1YB3 11824245 IC50 > 10000 nM T11388 CRXO59 11857300 IC50 = 3058 nM T11388 CDOG76 11857302 IC50 > 10000 nM T11388 CM0VY1 11957542 Ki = 1.4 nM T11388 C5NR3L 11962098 IC50 < 1 nM T11388 C3QN1E 11983275 Ki = 1.7 nM T11388 C89TXY 11990595 IC50 = 0.62 nM T11388 CFK68L 12414738 IC50 = 4780 nM T11388 CHW30V 12967046 IC50 = 1.18 ug.mL-1 T11388 C31MCN 13186896 IC50 > 100000 nM T11388 CT2J7M 13245620 IC50 = 78 nM T11388 CD4V3O 13820370 IC50 = 540 nM T11388 C4JQR9 14060550 Ki > 1000000 nM T11388 COP0K2 14308232 Ki > 1000000 nM T11388 C9WC6M 14655218 Ki = 260 nM T11388 CM7H4S 15283376 Ki = 136000 nM T11388 CV3AR1 15345958 Ki = 3.5 nM T11388 CN91PY 15547226 IC50 > 2500 nM T11388 CCGS52 15547237 IC50 = 2.5 nM T11388 CLGV32 15547238 IC50 = 100 nM T11388 CI8QZ5 15567852 Ki > 1000000 nM T11388 CVO9K6 15858812 IC50 = 1630 nM T11388 CHC31Q 15985697 IC50 = 0.6 nM T11388 C8A7ER 15985701 IC50 = 0.2 nM T11388 C9LW6H 15985754 IC50 = 0.6 nM T11388 CAY67P 15992537 IC50 > 30000 nM T11388 CQ5F9T 16045426 IC50 = 0.2 nM T11388 CO6B8V 16046088 IC50 = 67 nM T11388 CL38RU 16046125 Ki > 100000 nM T11388 CQ2N8D 16046128 Ki > 30000 nM T11388 C08XJK 16090559 Ki = 880 nM T11388 CTIV96 16090560 Ki = 430 nM T11388 C2QWA9 16090561 Ki > 10000 nM T11388 CJBT92 16090562 Ki = 1700 nM T11388 CU6KB8 16090563 Ki > 15000 nM T11388 CM1S0X 16108886 IC50 > 1000 nM T11388 CZ9J6G 16108888 IC50 = 0.022 nM T11388 C3KMJ0 16108889 IC50 = 0.75 nM T11388 CM7DA6 16108890 IC50 < 0.003 nM T11388 C0M1KY 16108891 IC50 < 0.003 nM T11388 C63XFT 16108892 IC50 = 0.025 nM T11388 C0LJ8Y 16108893 IC50 = 0.011 nM T11388 C7IQ0W 16108894 IC50 = 0.003 nM T11388 CPN5S2 16108895 IC50 = 0.031 nM T11388 CH2SV7 16108898 IC50 > 1000 nM T11388 CJ98LN 16108900 IC50 = 10 nM T11388 CYT2X8 16108901 IC50 = 0.009 nM T11388 CJRB12 16108902 IC50 = 0.047 nM T11388 C0QAC5 16108903 IC50 = 0.3 nM T11388 CT65ZO 16108904 IC50 = 0.011 nM T11388 CHKR18 16108905 IC50 = 0.013 nM T11388 CZI27Q 16108906 IC50 = 0.003 nM T11388 C6D4FQ 16655063 IC50 = 3.8 nM T11388 CHR1G5 16661368 IC50 = 174 nM T11388 C5FUL9 16661369 IC50 = 238 nM T11388 CUTI57 16661526 IC50 = 13 nM T11388 CEU86A 16661530 IC50 = 1045 nM T11388 C26JIW 16661682 IC50 = 10 nM T11388 C51WCU 16661683 IC50 = 6070 nM T11388 C8QD4E 16662142 IC50 = 8310 nM T11388 C6XPN4 16664855 IC50 = 38 nM T11388 C0QE5A 16666183 IC50 = 0.4 nM T11388 C8XLP2 16720100 Ki = 1240 nM T11388 C4P8ZV 16720327 Ki = 1280 nM T11388 CI0WO4 17747162 IC50 = 1660 nM T11388 CCPD37 17747164 IC50 = 447 nM T11388 CB7M2X 17747165 IC50 = 513 nM T11388 C9QRT6 17747166 IC50 = 270 nM T11388 CKA87T 17945762 IC50 = 51 nM T11388 CTQM93 17968180 IC50 = 4.7 nM T11388 CH4TC1 17968209 IC50 < 1 nM T11388 C0Q1ML 17968234 IC50 < 1 nM T11388 C0JBH9 18395047 IC50 = 2500 nM T11388 C2XTI9 18395048 IC50 = 2300 nM T11388 CLM87K 18537504 Ki = 13 nM T11388 C7WD4Z 18628647 IC50 = 97 nM T11388 CR7B9L 18628679 IC50 = 790 nM T11388 CHA0S3 18628693 IC50 = 18 nM T11388 CU3NM9 18628717 IC50 = 1227 nM T11388 C71IFZ 18628739 IC50 = 6 nM T11388 CUSD12 18628799 IC50 = 12 nM T11388 C34QUK 21309371 IC50 > 2500 nM T11388 C3Q0AW 22884155 IC50 = 51 nM T11388 C2KBL6 22972497 IC50 = 16 nM T11388 CD5R3V 22972573 IC50 = 37 nM T11388 CKW6Q8 23626706 IC50 = 405 nM T11388 CZ8DI1 23643986 Ki = 120 nM T11388 CCR95Y 23644161 IC50 = 0.25 nM T11388 CZ4T5P 23644230 IC50 = 26 nM T11388 C0QVL2 23644739 Ki = 125 nM T11388 CM1C8V 23644740 Ki > 30000 nM T11388 CM5TI6 23644741 Ki > 100000 nM T11388 CMQ72V 23644742 Ki > 100000 nM T11388 CZPF48 23648277 IC50 = 31 nM T11388 CHU59C 23648278 IC50 = 5 nM T11388 CA74XT 23648279 IC50 = 639 nM T11388 C2I6RW 23648280 IC50 = 5.3 nM T11388 CCJ8M5 23648281 IC50 = 1117 nM T11388 C9C0HK 23648282 IC50 = 314 nM T11388 CC50JD 23648283 IC50 = 141 nM T11388 CS1VW7 23648284 IC50 > 10000 nM T11388 CUQH43 23648285 IC50 > 10000 nM T11388 CM52JD 23648286 IC50 > 10000 nM T11388 CE09VM 23648287 IC50 > 10000 nM T11388 C1FRI4 23648288 IC50 > 10000 nM T11388 C9RNB7 23648289 IC50 = 305 nM T11388 C4J5MD 23648290 IC50 = 290 nM T11388 CY20DH 23648291 IC50 = 269 nM T11388 CF7O3H 23648292 IC50 = 376 nM T11388 CKI1W5 23648293 IC50 = 825 nM T11388 CN5S3K 23648294 IC50 = 314 nM T11388 CTB69E 23648295 IC50 = 691 nM T11388 C31XJH 23648296 IC50 = 4 nM T11388 C5ECI8 23648297 IC50 = 4123 nM T11388 CB7T3I 23648298 IC50 = 391 nM T11388 CVF2M6 23648299 IC50 = 6.7 nM T11388 CRZ56K 23648300 IC50 = 0.2 nM T11388 CQ1C8H 23648301 IC50 = 0.3 nM T11388 CQFD10 23648302 IC50 = 0.1 nM T11388 CFR23Q 23648303 IC50 = 0.3 nM T11388 C0FBS2 23648304 IC50 = 2.3 nM T11388 C67AYX 23648305 IC50 = 1.5 nM T11388 CN6R9M 23648306 IC50 = 2.6 nM T11388 C85PXH 23648308 IC50 = 1.2 nM T11388 CVH82R 23648309 IC50 < 0.2 nM T11388 COZK65 23648310 Ki = 43 nM T11388 CCF89E 23648311 Ki = 246 nM T11388 CS4NV6 23648312 Ki = 66 nM T11388 CC9S7T 23648313 Ki = 205 nM T11388 CCTK94 23648314 Ki > 100000 nM T11388 CG29HR 23648315 Ki > 30000 nM T11388 CY35VT 23648316 Ki = 123 nM T11388 CTX79K 23648317 Ki > 100000 nM T11388 C8T5FW 23648318 Ki > 100000 nM T11388 C02UQZ 23648319 Ki = 595 nM T11388 C1QVI4 23648320 Ki > 65000 nM T11388 CP4SY0 23648321 Ki > 100000 nM T11388 C9C7JR 23648322 Ki > 100000 nM T11388 CTY4J2 23648323 Ki > 100000 nM T11388 CGJ96H 23648326 Ki > 30000 nM T11388 CSI84Q 23648327 Ki > 100000 nM T11388 C2PD6A 23648328 Ki > 100000 nM T11388 C37FRY 23648329 Ki > 100000 nM T11388 C4KU8Q 23648330 Ki > 100000 nM T11388 C09TQZ 23648331 Ki > 100000 nM T11388 CM0AG6 23648332 Ki = 55 nM T11388 C8DJZ7 23648333 Ki = 58 nM T11388 CVH46G 23648334 Ki > 20000 nM T11388 C1IRW9 23648335 Ki > 100000 nM T11388 CWG7T3 23648336 Ki > 100000 nM T11388 CZN75B 23648337 Ki > 30000 nM T11388 CLZX16 23648338 Ki = 341 nM T11388 C5UDE3 23648339 Ki = 718 nM T11388 C7V6EY 23648340 Ki = 438 nM T11388 CRK1M0 23648341 Ki > 100000 nM T11388 C34VFB 23648342 Ki > 100000 nM T11388 CQUD83 23648343 Ki = 1581 nM T11388 C32GYK 23648344 Ki > 10000 nM T11388 CHQ82B 23648345 Ki = 131 nM T11388 CH0XM8 23648346 Ki = 125 nM T11388 C8ZT0W 23648347 Ki = 408 nM T11388 C5T6WQ 23648348 Ki = 478 nM T11388 CKE2C0 23648349 Ki = 310 nM T11388 CUH90V 23648350 Ki > 100000 nM T11388 CCA45G 23648351 Ki = 4320 nM T11388 CP10ST 23648352 Ki > 100000 nM T11388 CZRA72 23648353 Ki > 100000 nM T11388 CPTK56 23648354 Ki = 2750 nM T11388 C1YMU6 23648355 Ki = 47 nM T11388 C58JSH 23648356 Ki = 10760 nM T11388 C5YS0D 23648357 Ki > 100000 nM T11388 CNHA15 23648358 Ki = 55 nM T11388 CQVC57 23648359 Ki = 337 nM T11388 C03ZCQ 23648360 Ki > 100000 nM T11388 CM5QI0 23648361 Ki > 100000 nM T11388 C6YRH9 23648362 Ki > 100000 nM T11388 CP6Q2L 23648363 Ki = 2331 nM T11388 C63OZA 23648364 Ki > 100000 nM T11388 COU98B 23648365 Ki > 30000 nM T11388 CK43WQ 23648366 Ki = 2117 nM T11388 CKQ0P4 23648367 Ki > 100000 nM T11388 CGSN32 23648368 Ki > 100000 nM T11388 C76JKU 23648369 Ki > 100000 nM T11388 C46RQB 23648370 Ki > 30000 nM T11388 CPC7Z2 23648371 Ki > 30000 nM T11388 C5FJZ6 23648372 Ki > 30000 nM T11388 CL8X1T 23648373 Ki > 30000 nM T11388 CL01QA 23648374 Ki = 1390 nM T11388 CG9N8B 23648375 Ki = 1180 nM T11388 CT98GY 23648376 Ki = 3970 nM T11388 CX6JF9 23648377 Ki = 355 nM T11388 CJ7N9D 23648378 Ki > 100000 nM T11388 C0GQ4R 23648379 Ki > 30000 nM T11388 CYS7Z2 23648380 Ki > 30000 nM T11388 C6H3DY 23648381 Ki > 100000 nM T11388 CGV2J8 23648382 Ki > 100000 nM T11388 CF0JM1 23648383 Ki > 100000 nM T11388 C5LGJ7 23648384 Ki > 100000 nM T11388 C39FZB 23648385 Ki > 100000 nM T11388 C85STC 23648386 Ki > 100000 nM T11388 CWV98T 23648387 Ki > 100000 nM T11388 CX59EJ 23648388 Ki > 100000 nM T11388 CFNX14 23648389 Ki > 100000 nM T11388 CZC34G 23648390 Ki > 100000 nM T11388 C1FJY7 23648391 Ki = 8580 nM T11388 C9KW2O 23648392 Ki = 150 nM T11388 CI58TU 23648393 Ki > 30000 nM T11388 CB3JX0 23648394 Ki = 4610 nM T11388 CYBW67 23648395 Ki > 30000 nM T11388 CR1K4V 23648396 Ki > 30000 nM T11388 C1B9GH 23648397 Ki > 30000 nM T11388 CF72ZM 23648398 Ki > 30000 nM T11388 C9X3TS 23648399 Ki = 14300 nM T11388 CL8RT9 23648400 Ki = 13300 nM T11388 CPEW28 23648401 Ki = 1660 nM T11388 CT10OV 23648402 Ki = 130 nM T11388 CEC70K 23648403 Ki = 139 nM T11388 CE2QR4 23648404 Ki = 18800 nM T11388 C4F2BY 23648405 Ki > 100000 nM T11388 CX37JK 23648406 Ki = 1330 nM T11388 CD8JP5 23648407 Ki = 461 nM T11388 CC7HD5 23648408 Ki = 1540 nM T11388 CWGL69 23648409 Ki = 5130 nM T11388 CA2DE6 23648410 Ki = 13100 nM T11388 C3VT9K 23648411 Ki = 16900 nM T11388 CBR76L 23648414 IC50 = 48 nM T11388 CZ7ME6 23648415 IC50 = 120 nM T11388 CVU01O 23648416 IC50 = 63 nM T11388 C3M5GX 23648417 IC50 = 398 nM T11388 CG9NQ8 23648418 IC50 > 1000 nM T11388 C2F1MC 23648419 IC50 = 43 nM T11388 CCZ4J1 23648420 IC50 = 240 nM T11388 CC2W3A 23648421 IC50 = 9 nM T11388 C8Z5BC 23648422 IC50 = 83 nM T11388 CVD5Y6 23648423 IC50 = 9 nM T11388 CL4Q2D 23648424 IC50 < 1 nM T11388 CF0TY4 23648425 IC50 = 430 nM T11388 CX0V8M 23648426 IC50 < 1 nM T11388 CME4Y9 23648427 IC50 = 24 nM T11388 C4AJB0 23648428 IC50 = 190 nM T11388 CI1XK0 23648429 IC50 = 65 nM T11388 C6P3YR 23648430 IC50 = 18 nM T11388 C5AQX8 23648431 IC50 = 4 nM T11388 CQA3C5 23648432 IC50 = 300 nM T11388 CAS2L7 23648433 IC50 = 32 nM T11388 C0M8FS 23648434 IC50 = 6.4 nM T11388 CD7R1S 23648435 IC50 = 7.6 nM T11388 CF9H8N 23648436 IC50 = 5.5 nM T11388 CZG5U1 23648437 IC50 = 1.4 nM T11388 CF68MH 23648438 IC50 = 3.2 nM T11388 C9WS5T 23648439 IC50 > 250 nM T11388 C2C5YA 23648440 IC50 = 2.1 nM T11388 C7DBS2 23648441 Ki = 60 nM T11388 C0F1DO 23648442 Ki = 8 nM T11388 C4KS9Y 23648443 Ki = 560 nM T11388 CAUJ42 23648444 IC50 = 7.1 nM T11388 C1YTO9 23648449 IC50 = 1015 nM T11388 C2GQ6X 24897809 Ki = 0.064 nM T11388 CZ21HD 24898027 Ki = 0.14 nM T11388 CQU38W 24900755 IC50 = 553 nM T11388 C2S8VB 24901099 IC50 = 104 nM T11388 CIN28B 24901100 IC50 = 511 nM T11388 CD2EH0 24901101 IC50 = 1267 nM T11388 CS7B3F 24901102 IC50 > 10000 nM T11388 CG9H6V 25008106 IC50 = 69 nM T11388 CK7BR0 25023784 IC50 > 1500 nM T11388 CZH87T 25023785 IC50 = 5900 nM T11388 C2PUY3 25023786 IC50 > 1000 nM T11388 CFQM73 25023787 IC50 = 290 nM T11388 CTK09I 25023788 IC50 = 79 nM T11388 CDL98C 25023789 IC50 > 1000 nM T11388 CCP3G0 25023790 IC50 > 2000 nM T11388 CGI0U2 25023791 IC50 = 5400 nM T11388 CO72TX 25027584 IC50 = 100 nM T11388 CMS0L3 25052748 IC50 > 1000 nM T11388 C7J3MN 25053851 IC50 < 1 nM T11388 C6AVL9 25053852 IC50 < 1 nM T11388 C19GML 25071954 IC50 = 44 nM T11388 CF54QZ 25129041 IC50 = 50.12 nM T11388 CDO26T 25129042 IC50 = 10 nM T11388 C57LJM 25129043 IC50 = 3 nM T11388 C3AT6W 25130088 IC50 = 8 nM T11388 C1FWI6 25133836 IC50 = 18 nM T11388 CYV1J6 25133837 IC50 = 312 nM T11388 CBZK08 25133838 IC50 = 12.59 nM T11388 CP8U3Q 25142042 IC50 < 1 nM T11388 CC92AI 25142043 IC50 < 1 nM T11388 C8IFW0 25142172 IC50 = 3 nM T11388 CD2A6W 25142173 IC50 = 1 nM T11388 C53OMA 25142175 IC50 = 3 nM T11388 C7CFR2 25142176 IC50 = 42 nM T11388 C78RJG 25142177 IC50 = 41 nM T11388 CS6R4T 25142308 IC50 = 50 nM T11388 CM2PI4 25142309 IC50 = 10 nM T11388 CM6FL3 25142310 IC50 = 4 nM T11388 CWV4F5 25142312 IC50 = 4 nM T11388 CH52AJ 25142313 IC50 = 78 nM T11388 COG9V7 25142440 IC50 < 1 nM T11388 CYL56K 25142444 IC50 = 2 nM T11388 C3IT4O 25142445 IC50 = 2 nM T11388 CK7D0V 25142571 IC50 = 4 nM T11388 CW9KR5 25142573 IC50 = 2 nM T11388 CZ0G2I 25142574 IC50 < 1 nM T11388 CNH31I 25142699 IC50 = 5 nM T11388 CQ9PD6 25142700 IC50 = 17 nM T11388 CV08DB 25142970 IC50 = 34 nM T11388 C3C8YJ 25174148 IC50 = 39.81 nM T11388 C5M1BT 25195691 IC50 = 251.19 nM T11388 CTLO73 25204268 IC50 = 871 nM T11388 C42ZMF 25204335 IC50 = 468 nM T11388 CC7TV3 25204336 IC50 = 331 nM T11388 CFX41G 25204403 IC50 = 2291 nM T11388 CU59SO 25242431 Ki = 1800 nM T11388 C23JPC 25242432 Ki = 270 nM T11388 CW9JM2 25256832 IC50 = 18 nM T11388 C3GC7P 25256833 IC50 = 6 nM T11388 CB4P0U 40495533 IC50 > 30000 nM T11388 CZS24P 42633520 IC50 = 3 nM T11388 CI78XT 42633521 IC50 = 2 nM T11388 CZ6B1F 42635119 IC50 = 0.9 nM T11388 CZM36T 42641892 IC50 = 1000 nM T11388 CRYH80 42642459 IC50 = 398.11 nM T11388 C3DC4M 42647278 Ki = 2 nM T11388 C25ELB 44143088 IC50 = 23.44 nM T11388 C9QDC0 44143091 IC50 = 50.12 nM T11388 CNM6X8 44218399 IC50 = 25 nM T11388 CJA68L 44224113 IC50 = 3162.28 nM T11388 C2V5ZT 44224114 IC50 > 10000 nM T11388 C0U9VJ 44224115 IC50 > 10000 nM T11388 C0MZ9D 44224116 IC50 = 5011.87 nM T11388 CEJ82A 44224117 IC50 = 1258.93 nM T11388 C0KL7D 44224118 IC50 = 6309.57 nM T11388 CE9S0M 44224119 IC50 = 5011.87 nM T11388 CV1W0Z 44224120 IC50 = 6309.57 nM T11388 C5LDK7 44224121 IC50 = 6309.57 nM T11388 C8UF5Q 44224122 IC50 > 10000 nM T11388 C9YHC5 44224123 IC50 = 5011.87 nM T11388 CA26RI 44224124 IC50 > 10000 nM T11388 CU0PI2 44224125 IC50 > 10000 nM T11388 CRL79W 44224126 IC50 > 10000 nM T11388 C3T0QO 44224127 IC50 > 10000 nM T11388 C81EVM 44224128 IC50 = 2511.89 nM T11388 C7IY8P 44224129 IC50 = 6309.57 nM T11388 CYG02V 44224130 IC50 = 10000 nM T11388 CJS1B9 44224131 IC50 = 1258.93 nM T11388 CN5O8S 44224132 IC50 = 5011.87 nM T11388 C2Q3RP 44224133 IC50 = 5011.87 nM T11388 CZX62T 44224134 IC50 = 1995.26 nM T11388 CP3YA9 44224135 IC50 = 3162.28 nM T11388 CSZH31 44224136 IC50 = 2511.89 nM T11388 CT7VX0 44279004 Ki = 30 nM T11388 CR38EU 44279051 Ki = 2 nM T11388 C5LJS7 44279083 Ki = 2.6 nM T11388 C2V7RL 44279437 Ki = 2.3 nM T11388 CD84XF 44279475 IC50 = 72 nM T11388 C0RQ3V 44279712 IC50 = 16 nM T11388 CFJ2Z1 44279771 IC50 = 100 nM T11388 C3IBQ0 44279792 IC50 = 2500 nM T11388 CQ57HR 44279823 IC50 = 100 nM T11388 C5YF0J 44279873 IC50 > 5000 nM T11388 C6ZXK0 44280152 IC50 = 100 nM T11388 CVZ54E 44280172 IC50 = 38 nM T11388 CHPM71 44299700 Ki = 330 nM T11388 CO8PZ6 44302078 Ki = 38 nM T11388 C1UW0M 44302097 Ki = 180 nM T11388 CUGK48 44302128 Ki > 10000 nM T11388 C6SA2N 44302130 Ki > 10000 nM T11388 CNPF54 44302142 Ki > 10000 nM T11388 CQ2O7B 44302157 Ki = 420 nM T11388 CKPF47 44302158 Ki = 61 nM T11388 CP0F7Z 44302170 Ki = 190 nM T11388 CK0GS8 44302171 Ki > 10000 nM T11388 C3U7GN 44302172 Ki > 10000 nM T11388 CD2Q5Y 44302173 Ki > 10000 nM T11388 CYZ5I8 44302222 Ki > 10000 nM T11388 CS4K7I 44302226 Ki > 10000 nM T11388 C1I7FR 44302259 Ki > 10000 nM T11388 CKV9Z4 44302280 Ki > 10000 nM T11388 CZKU93 44302325 Ki > 1000 nM T11388 C8U3MI 44302326 Ki = 64 nM T11388 CI6NU5 44302384 Ki = 820 nM T11388 CL43BW 44302477 Ki = 53 nM T11388 C4KPU5 44302478 Ki = 640 nM T11388 C9WP1M 44302500 Ki = 11 nM T11388 CG67PQ 44302501 Ki > 1000 nM T11388 CN96YS 44302523 Ki = 710 nM T11388 CK1GD6 44302524 Ki > 1000 nM T11388 CNL8Y4 44302956 IC50 = 419 nM T11388 CAM2S5 44302974 IC50 = 280 nM T11388 CBYD40 44302975 IC50 < 3 nM T11388 CNA24Z 44303031 IC50 = 36 nM T11388 C56IEO 44303058 IC50 = 43 nM T11388 CL4VM1 44303061 IC50 = 49 nM T11388 CU9I1M 44303247 Ki = 10 nM T11388 CV7E9M 44303265 Ki = 32 nM T11388 C7RI3A 44303267 Ki = 15 nM T11388 CS0P5A 44303274 IC50 > 1000 nM T11388 CXU16T 44303285 IC50 = 81 nM T11388 CEIH70 44303290 IC50 > 1000 nM T11388 CN21AS 44303309 IC50 = 855 nM T11388 C24EDH 44303315 IC50 = 1000 nM T11388 CDX5M7 44303318 IC50 = 4 nM T11388 CRK48P 44303319 IC50 = 3 nM T11388 CKB9O1 44303324 IC50 < 3 nM T11388 C0FEJ1 44303335 IC50 = 44 nM T11388 CT49MJ 44303338 IC50 = 490 nM T11388 CMF6W2 44303344 IC50 < 3 nM T11388 CD1HJ5 44303345 IC50 < 3 nM T11388 CL26OE 44303389 IC50 < 30 nM T11388 CN9QY5 44303414 IC50 = 152 nM T11388 CRAB46 44303553 Ki = 7 nM T11388 CQCZ32 44303601 Ki = 470 nM T11388 CYAF19 44303687 Ki = 590 nM T11388 C4ZMH3 44303688 Ki = 68 nM T11388 CG3OM8 44304535 Ki = 380 nM T11388 C0FKB3 44304563 Ki = 160 nM T11388 CC04TQ 44304591 Ki = 950 nM T11388 C76OIY 44304610 Ki = 8.8 nM T11388 CK8JW5 44304611 Ki = 200 nM T11388 CZ87NW 44304634 Ki = 2100 nM T11388 COR96D 44304861 Ki = 3600 nM T11388 CNWP14 44319207 IC50 = 18000 nM T11388 CAE2M6 44319219 IC50 = 13000 nM T11388 CVH6I8 44319220 IC50 = 1000 nM T11388 CAC20W 44319316 IC50 = 23000 nM T11388 CI6QO0 44319483 IC50 = 59000 nM T11388 CM95NF 44319484 IC50 = 44000 nM T11388 CF8V1M 44319498 IC50 = 30000 nM T11388 CY81RN 44319518 IC50 = 14000 nM T11388 C9O1VP 44319528 Ki = 683 nM T11388 CO7NB1 44319649 IC50 = 19000 nM T11388 CH9E6N 44321598 Ki = 1370 nM T11388 C6EYQ8 44321883 Ki = 229 nM T11388 CTW41Y 44321884 Ki = 1061 nM T11388 CU7J2P 44321946 Ki = 492 nM T11388 CKU37V 44326283 IC50 = 23 nM T11388 CB80NG 44326383 IC50 = 83 nM T11388 C36NXS 44326384 IC50 = 660 nM T11388 C27WCO 44326483 IC50 = 50 nM T11388 CXWY65 44326484 IC50 = 41 nM T11388 C79QSL 44326485 IC50 = 29 nM T11388 CFI1T7 44326490 IC50 = 98 nM T11388 C4PE9H 44326517 IC50 = 680 nM T11388 C62IYX 44326653 IC50 = 130 nM T11388 CN67DH 44326654 IC50 = 110 nM T11388 CL7HV3 44326812 IC50 = 250 nM T11388 C8R5MK 44326855 IC50 = 87 nM T11388 CT3RM0 44326856 IC50 = 26 nM T11388 CK20WD 44326888 IC50 = 410 nM T11388 C0M1TB 44326889 IC50 = 150 nM T11388 C4D1PT 44326891 IC50 = 41 nM T11388 CRM10A 44326910 IC50 = 15 nM T11388 C3UKH4 44326942 IC50 = 370 nM T11388 C9YWU3 44326970 IC50 = 79 nM T11388 CW6GY3 44326971 IC50 = 15 nM T11388 C0MF5A 44329571 Ki = 1440 nM T11388 CKB02C 44329582 Ki = 1000 nM T11388 CTN34G 44329585 Ki = 20 nM T11388 CR1J6F 44329593 Ki = 67 nM T11388 C3EHF1 44329596 Ki = 111 nM T11388 C97WPV 44329608 Ki = 110 nM T11388 CY5KH4 44329643 Ki = 947 nM T11388 CD24MB 44331308 IC50 = 590 nM T11388 C0AP9X 44331713 IC50 = 780 nM T11388 C78KLP 44331734 IC50 = 280 nM T11388 CGSO26 44331735 IC50 = 700 nM T11388 CSE71X 44331754 IC50 = 1400 nM T11388 CV28OM 44331755 IC50 = 740 nM T11388 C2EC3S 44331756 IC50 = 590 nM T11388 CL0Z2K 44331787 IC50 = 840 nM T11388 CLC86R 44331797 IC50 = 1500 nM T11388 C7MWQ8 44342499 IC50 = 6 nM T11388 CQ61OB 44342501 IC50 = 2500 nM T11388 CIBF96 44342511 IC50 = 1.8 nM T11388 CVK4H3 44342519 IC50 = 400 nM T11388 CN7BH9 44342744 IC50 > 2500 nM T11388 CP2OM5 44342745 IC50 = 7.6 nM T11388 CMQ6Y0 44342776 IC50 = 100 nM T11388 CHP3M7 44342892 IC50 = 71 nM T11388 CAF06H 44342893 IC50 = 6.5 nM T11388 C2CEM5 44342960 IC50 = 5 nM T11388 C6PLY0 44342983 IC50 = 35 nM T11388 CSQU25 44343007 IC50 = 4.6 nM T11388 C1IJW5 44343023 IC50 = 2 nM T11388 CO1K4S 44343024 IC50 = 7.6 nM T11388 CSBK92 44343025 IC50 = 1.5 nM T11388 C71JRX 44343028 IC50 = 0.13 nM T11388 COEK09 44343037 IC50 = 2.7 nM T11388 C0VF8I 44343038 IC50 = 100 nM T11388 C6Y4IQ 44343046 IC50 = 4 nM T11388 C27GXO 44343068 IC50 = 3.1 nM T11388 C61UIS 44343092 IC50 = 2.1 nM T11388 C4TLY5 44343100 IC50 = 600 nM T11388 CB64RL 44343105 IC50 = 2.4 nM T11388 C4YO9N 44343106 IC50 = 12 nM T11388 C4LBU1 44343120 IC50 = 270 nM T11388 CN0F3P 44343178 IC50 = 2.9 nM T11388 C0JBT1 44343179 IC50 = 5.4 nM T11388 C2MXH1 44343180 IC50 = 4.7 nM T11388 C8PQH2 44343355 IC50 = 1.1 nM T11388 C9OKX2 44343356 IC50 = 0.56 nM T11388 C9EB0F 44343357 IC50 = 0.87 nM T11388 C0TAX2 44345292 Ki = 30 nM T11388 CD9P4K 44345387 Ki = 900 nM T11388 C8HP5M 44347822 IC50 = 10 nM T11388 CK0B9C 44347827 IC50 = 2580 nM T11388 CO82ZV 44347993 IC50 = 630 nM T11388 CLCP51 44348116 IC50 = 614 nM T11388 CFBI42 44348134 IC50 = 150 nM T11388 CYEI89 44348185 IC50 = 58 nM T11388 CGF04H 44348385 IC50 = 3 nM T11388 C9PZ5H 44370493 IC50 = 87 nM T11388 CLES53 44375718 IC50 = 5900 nM T11388 C76OGS 44375719 IC50 > 100000 nM T11388 CA3E5V 44375741 IC50 = 2884.03 nM T11388 C31RPH 44375755 IC50 = 9100 nM T11388 CHL7A5 44375756 IC50 = 21000 nM T11388 C7QZ0F 44375757 IC50 = 18197.01 nM T11388 CEK1B0 44375761 IC50 = 0.79 nM T11388 CS0TA4 44375775 IC50 = 912.01 nM T11388 CIEQ12 44375794 IC50 = 1.096 nM T11388 C5RGE9 44375809 IC50 = 33.88 nM T11388 CKNR62 44375810 IC50 = 3388.44 nM T11388 CYN84V 44375815 IC50 = 1200 nM T11388 CY3S7H 44375830 IC50 = 19.95 nM T11388 CRWF03 44375905 IC50 = 6.31 nM T11388 CT92UX 44375906 IC50 = 69 nM T11388 C45PSC 44375926 IC50 = 0.7079 nM T11388 CYAB62 44375947 IC50 = 4168.69 nM T11388 CC24WK 44375966 IC50 = 5000 nM T11388 CV80FS 44375983 IC50 = 6300 nM T11388 CR31GV 44376125 IC50 = 76 nM T11388 CZA2X4 44376143 IC50 > 100000 nM T11388 C3KR5O 44376144 IC50 = 32 nM T11388 CWCZ58 44376146 IC50 = 1400 nM T11388 CA9LC3 44382185 Ki = 14 nM T11388 C5NH3W 44382186 Ki = 8 nM T11388 CZU70X 44382187 Ki = 3 nM T11388 C3M5CT 44382237 Ki = 3 nM T11388 C3W7CI 44382238 Ki = 4 nM T11388 CM9WG5 44382239 Ki = 706 nM T11388 CUEX04 44382949 Ki = 12 nM T11388 C9UQN0 44383254 Ki > 10000 nM T11388 CU4CB8 44383255 Ki = 9 nM T11388 C83ART 44383306 Ki = 5 nM T11388 CEUA60 44383413 Ki = 15 nM T11388 CX20UA 44383464 Ki = 1100 nM T11388 C12AOQ 44389682 Ki = 4.8 nM T11388 CC6VR0 44391415 IC50 = 300 nM T11388 C5M0AT 44391418 IC50 = 19 nM T11388 CEYK19 44391428 IC50 = 380 nM T11388 CJ76PM 44391433 IC50 = 8100 nM T11388 CNF0V9 44391443 IC50 > 1300 nM T11388 CMRH32 44391458 IC50 > 1300 nM T11388 CP7KW2 44391459 Ki = 1.8 nM T11388 C9W3HN 44391474 IC50 = 0.048 nM T11388 CV71WQ 44391475 IC50 = 12 nM T11388 CR86LD 44391478 IC50 = 430 nM T11388 C8LYI2 44391485 IC50 = 8.9 nM T11388 CA39NJ 44391490 IC50 = 60 nM T11388 CD06XO 44391491 IC50 = 200 nM T11388 CXL54A 44391513 IC50 > 13000 nM T11388 CM71QV 44391553 IC50 = 1900 nM T11388 CLDX72 44391556 IC50 = 13000 nM T11388 C9URV1 44391588 IC50 = 13000 nM T11388 CL4P9T 44391610 IC50 = 7100 nM T11388 CXSR60 44391614 IC50 = 4000 nM T11388 C0EVK9 44391616 IC50 = 8100 nM T11388 CJ8X0Q 44391624 IC50 = 3100 nM T11388 CBC4G3 44391705 IC50 > 13000 nM T11388 CTRP74 44394287 IC50 = 65 nM T11388 CP7X6J 44394353 IC50 = 12.88 nM T11388 C4M3EN 44394384 IC50 = 7.6 nM T11388 CQL46I 44394417 IC50 = 24 nM T11388 C79NFU 44394458 IC50 = 25 nM T11388 CQD39O 44394488 IC50 = 710 nM T11388 C1E3YD 44394519 IC50 = 630 nM T11388 CUZ30C 44394534 IC50 = 150 nM T11388 C1HDY3 44396728 IC50 = 5.5 nM T11388 CV18UI 44396786 IC50 = 7.9 nM T11388 C2J6MW 44397423 IC50 = 650 nM T11388 CRSF50 44397609 IC50 = 0.3388 nM T11388 CHWX97 44397693 IC50 = 2.818 nM T11388 CZC50Y 44398247 IC50 >> 1000 nM T11388 CQPM06 44398248 IC50 >> 1000 nM T11388 CYJ8Z4 44398353 IC50 = 10 nM T11388 CD73QR 44398649 Ki = 0.019 nM T11388 CXOU54 44398650 Ki = 1500 nM T11388 CHQF16 44398651 Ki = 0.009 nM T11388 C4ALQ9 44398659 Ki = 26 nM T11388 CA5S6C 44398660 Ki = 2300 nM T11388 CI5TK4 44398665 Ki = 830 nM T11388 CVF5Q3 44398666 Ki = 0.007 nM T11388 C6YP7B 44398667 Ki = 0.006 nM T11388 C5MDW7 44398676 Ki = 0.003 nM T11388 C4D9MO 44398688 Ki = 7900 nM T11388 CUW76J 44398689 Ki > 13000 nM T11388 CXY3H0 44398710 Ki > 13000 nM T11388 CGQ20I 44398741 Ki = 0.032 nM T11388 CW2YL6 44398760 Ki = 0.004 nM T11388 CDZA87 44398761 Ki = 0.004 nM T11388 CCAV34 44398779 Ki > 13000 nM T11388 C20FET 44398780 Ki = 62 nM T11388 CD18YP 44402055 IC50 = 32 nM T11388 CU8TB9 44402056 IC50 = 7.2 nM T11388 CD4TP7 44402158 IC50 = 100 nM T11388 CO6BG2 44402160 IC50 = 5.7 nM T11388 C0AJC4 44402175 IC50 = 190 nM T11388 CX9O2Q 44402263 IC50 = 350 nM T11388 C89MOT 44402291 IC50 = 26 nM T11388 CFL9B8 44402952 IC50 = 4.6 nM T11388 CRZT97 44403028 IC50 = 5 nM T11388 CTX0C1 44403029 IC50 = 802 nM T11388 CPS6Z4 44403032 IC50 = 988 nM T11388 CB1Q8T 44403033 IC50 = 2.4 nM T11388 C3Z0AJ 44403034 IC50 = 2.5 nM T11388 CJ0K5D 44403035 IC50 = 30 nM T11388 CW2L5D 44404573 Ki > 100000 nM T11388 C39PTS 44404574 Ki > 100000 nM T11388 C9FXS8 44406940 IC50 = 1.7 nM T11388 C3D1CO 44406943 IC50 = 4.2 nM T11388 C7IHW3 44406951 IC50 = 0.5 nM T11388 C1R6VD 44407011 IC50 = 0.58 nM T11388 C9YS7A 44407059 IC50 = 280 nM T11388 CJ9Z2O 44407919 IC50 = 490 nM T11388 CIM1N8 44407924 IC50 = 170 nM T11388 C9G4NY 44407925 IC50 = 160 nM T11388 COR8Q5 44407926 IC50 = 400 nM T11388 CB3KR0 44407927 IC50 = 410 nM T11388 CZG60N 44407947 IC50 = 260 nM T11388 CFXQ80 44407948 IC50 = 180 nM T11388 CQU10Z 44407969 IC50 = 350 nM T11388 C7M8WH 44407970 IC50 = 280 nM T11388 CK9NV4 44408004 IC50 = 1100 nM T11388 CWVN14 44408009 IC50 = 520 nM T11388 C4ZMP9 44408016 IC50 = 35 nM T11388 CG1RT6 44408023 IC50 = 830 nM T11388 CIOJ71 44408024 IC50 = 200 nM T11388 CBD8R9 44408038 IC50 = 220 nM T11388 CTX29M 44408043 IC50 = 24 nM T11388 CKM7Y2 44408044 IC50 = 130 nM T11388 C25RIN 44408049 IC50 = 0.33 nM T11388 CD4T1S 44408059 IC50 = 93 nM T11388 CO5BW8 44408060 IC50 = 31 nM T11388 CNQ5X3 44408079 IC50 = 170 nM T11388 C7QLA3 44408090 IC50 = 72 nM T11388 CCW4V2 44408091 IC50 = 40 nM T11388 CN6U8E 44408092 IC50 = 36 nM T11388 CLX20F 44408094 IC50 = 470 nM T11388 CX26IH 44408095 IC50 = 45 nM T11388 C4EBJ3 44408098 IC50 = 58 nM T11388 CFKB96 44408101 IC50 = 11000 nM T11388 CHIG10 44408102 IC50 = 520 nM T11388 CV85CH 44408112 IC50 = 470 nM T11388 CAR54M 44408113 IC50 = 33000 nM T11388 C57VLN 44408673 IC50 = 3000 nM T11388 C7MG9V 44408680 IC50 = 10 nM T11388 C12SFP 44408699 IC50 = 1200 nM T11388 C51TZE 44408700 IC50 = 90 nM T11388 CP8E9I 44408704 IC50 = 100 nM T11388 C1NG6B 44408705 IC50 > 20000 nM T11388 C8CXU5 44408707 IC50 = 83 nM T11388 CQPW10 44408746 IC50 = 69 nM T11388 CVA6D2 44408747 IC50 = 600 nM T11388 CODU85 44408752 IC50 = 100 nM T11388 CZ2BQ0 44408754 IC50 = 40 nM T11388 CL3K0B 44408758 IC50 = 60 nM T11388 C7BGH5 44408774 IC50 = 11 nM T11388 C79CUE 44408891 IC50 = 3000 nM T11388 CCD39H 44408906 IC50 = 99 nM T11388 C6MOX3 44408907 IC50 = 11000 nM T11388 C1FMZ0 44408912 IC50 = 82 nM T11388 CR3Q4S 44408934 IC50 = 320 nM T11388 CM7FI3 44408935 IC50 = 190 nM T11388 C3RAF2 44408939 IC50 = 130 nM T11388 CWS86M 44408945 IC50 = 10 nM T11388 C51TCA 44408976 IC50 = 200 nM T11388 C9IEW7 44409018 Ki = 184 nM T11388 CX14BH 44409362 IC50 = 4.3 nM T11388 CT8G9X 44409364 IC50 = 17 nM T11388 CUBF53 44409368 IC50 = 24 nM T11388 C4PI7L 44409371 IC50 = 3.8 nM T11388 CVK3N9 44409380 IC50 = 2.8 nM T11388 CT1Q8S 44409384 IC50 = 27 nM T11388 C1G5JE 44409386 IC50 = 16 nM T11388 CREG93 44409399 IC50 = 1.7 nM T11388 CQ6HG4 44409402 IC50 = 6.9 nM T11388 CG5TS8 44409403 IC50 = 58 nM T11388 C0LDH2 44409407 IC50 = 5 nM T11388 CPM27T 44409408 IC50 = 2.1 nM T11388 CCN4Y1 44409411 IC50 = 32 nM T11388 CDS9E4 44409416 IC50 = 2.1 nM T11388 CIDV28 44409417 IC50 = 1.6 nM T11388 C1VTZ9 44409424 IC50 = 21 nM T11388 CI1C7Y 44409425 IC50 = 6.6 nM T11388 CU89IS 44409426 IC50 = 65 nM T11388 CX4ML9 44409428 IC50 = 8.3 nM T11388 CJY17B 44409432 IC50 = 3 nM T11388 CA58KV 44409435 IC50 = 29 nM T11388 CVW5I8 44409438 IC50 = 0.42 nM T11388 CD1Y7P 44409439 IC50 = 0.81 nM T11388 CKVF42 44409440 IC50 = 1 nM T11388 C6YEU9 44409449 IC50 = 8.9 nM T11388 C5X8AO 44409450 IC50 = 14 nM T11388 C0D4PK 44409451 IC50 = 15 nM T11388 CY4H2I 44411981 Ki < 0.25 nM T11388 CNU4T9 44412155 Ki < 0.25 nM T11388 CYF1B9 44412339 Ki = 17000 nM T11388 C1J6OW 44412340 Ki = 5600 nM T11388 CU49OM 44412341 Ki = 810 nM T11388 CDK32G 44412349 Ki = 35 nM T11388 CL82XD 44412354 Ki = 9600 nM T11388 C23ZVR 44412355 Ki = 3000 nM T11388 CV26BC 44412365 Ki = 500 nM T11388 CX93NW 44412366 Ki = 120 nM T11388 CZN9T0 44412387 Ki = 3.3 nM T11388 CY90QW 44412402 Ki = 5.2 nM T11388 C1HW8F 44412424 Ki = 19 nM T11388 CYDJ14 44412436 Ki = 0.95 nM T11388 CV49GB 44412437 Ki = 52000 nM T11388 CZ5VW2 44412440 Ki = 43 nM T11388 CZR1O3 44412502 Ki = 33000 nM T11388 CA23SL 44414977 Ki = 3.5 nM T11388 C0XB2M 44414978 Ki = 1.3 nM T11388 CAG5F3 44414992 Ki = 4.8 nM T11388 C8JL9C 44415006 Ki = 3 nM T11388 CZP7F3 44420106 IC50 = 0.77 ug.mL-1 T11388 CS6X7V 44426055 IC50 = 1833 nM T11388 C8IB2W 44426056 IC50 > 100000 nM T11388 CWL7D5 44440441 IC50 = 2 nM T11388 C7DBR1 44440443 IC50 = 1 nM T11388 C89JFL 44440444 IC50 = 1 nM T11388 C6JRX3 44440447 IC50 = 5 nM T11388 C7J8TZ 44440448 IC50 = 8 nM T11388 C9O8JR 44440450 IC50 = 4 nM T11388 C4TJ7U 44440451 IC50 = 2 nM T11388 CL09FQ 44440453 IC50 = 0.2 nM T11388 CGV87Y 44440454 IC50 = 0.4 nM T11388 CXW8C5 44442251 IC50 = 66 nM T11388 CI1KS2 44442252 IC50 = 109 nM T11388 C7X3FM 44442255 IC50 = 151 nM T11388 CP0S4Z 44442256 IC50 = 273 nM T11388 CVD7L4 44442257 IC50 = 1.2 nM T11388 C9MS5I 44442264 IC50 = 41 nM T11388 C60XDN 44442265 IC50 = 27 nM T11388 CF3B7G 44442266 IC50 = 120 nM T11388 CA10YS 44442267 IC50 = 87 nM T11388 C21KGX 44442268 IC50 = 277 nM T11388 CCX07D 44442269 IC50 = 238 nM T11388 CFN67O 44444198 IC50 = 15 nM T11388 C24AIO 44444199 IC50 = 2.3 nM T11388 CCM4R1 44444200 IC50 = 47 nM T11388 CR3DP0 44444201 IC50 = 3.4 nM T11388 CN5OJ8 44444202 IC50 = 1.5 nM T11388 CRJ07X 44444203 IC50 = 1.2 nM T11388 CSUC26 44444204 IC50 < 1 nM T11388 C3J4DH 44444205 IC50 < 1 nM T11388 C5T1NC 44444208 IC50 = 1 nM T11388 CGCU82 44444211 IC50 = 1.1 nM T11388 CGB81X 44444216 IC50 < 1 nM T11388 C9VB5M 44444217 IC50 < 1 nM T11388 C8FN2V 44444218 IC50 < 1 nM T11388 C1L9BM 44444221 IC50 < 1 nM T11388 CZ25FP 44444222 IC50 < 1 nM T11388 CTW39N 44444223 IC50 < 1 nM T11388 C6J8LS 44444224 IC50 = 1.1 nM T11388 CW2L4V 44444225 IC50 < 1 nM T11388 CA9JR0 44444228 IC50 < 1 nM T11388 CTQ81M 44444229 IC50 < 1 nM T11388 CWE50F 44444230 IC50 < 1 nM T11388 CT8QV6 44444231 IC50 = 4 nM T11388 CISQ24 44444232 IC50 = 5 nM T11388 C8CQS6 44444233 IC50 = 4 nM T11388 CP79CA 44444234 IC50 = 1 nM T11388 CXO56L 44447657 IC50 = 5.1 nM T11388 CB6H5U 44447658 IC50 = 4 nM T11388 C1U6JA 44447659 IC50 = 0.3 nM T11388 CV3T1A 44447660 IC50 = 16 nM T11388 CF7AV1 44447661 IC50 = 0.3 nM T11388 C7HRP2 44447662 IC50 = 0.4 nM T11388 C0CZ7P 44447663 IC50 = 0.2 nM T11388 CAF54M 44447664 IC50 < 0.2 nM T11388 CC4J7S 44447665 IC50 = 1.5 nM T11388 CL6WZ1 44450271 IC50 = 7.1 nM T11388 C3B2TR 44450349 IC50 = 4.8 nM T11388 C38JBH 44450361 IC50 = 19 nM T11388 CC0AG3 44452909 Ki = 40 nM T11388 CB8IX2 44452912 Ki = 8.5 nM T11388 CXJF30 44452936 Ki = 9.5 nM T11388 CVCJ36 44452938 Ki < 0.25 nM T11388 C4ZBF6 44452963 Ki = 3000 nM T11388 CWCK10 44452964 Ki = 500 nM T11388 CF9PC3 44452965 Ki = 9600 nM T11388 C8Z4WO 44459967 IC50 = 17.38 nM T11388 C86ORE 44459987 IC50 = 20.42 nM T11388 C9TFJ8 44464926 IC50 = 79.43 nM T11388 CYO0T1 44465454 IC50 = 7.943 nM T11388 CE83YL 44465721 IC50 = 1.995 nM T11388 CVD48M 44478848 IC50 = 4 nM T11388 CJR45G 44479122 IC50 = 6 nM T11388 C8I9QK 44479381 IC50 = 24 nM T11388 CWS3K7 44479385 IC50 = 11 nM T11388 C2PK4G 44479635 IC50 = 23 nM T11388 CB73NC 44479637 IC50 = 1 nM T11388 CFYP92 44482496 IC50 = 55 nM T11388 CQ4S7Y 44565776 IC50 = 110 nM T11388 CH8A2V 44565777 IC50 = 560 nM T11388 C30GNW 44565778 IC50 = 13 nM T11388 CCX8F0 44565779 IC50 = 23 nM T11388 CV1IL5 44565796 IC50 = 17 nM T11388 C6MKC1 44565797 IC50 = 300 nM T11388 C1BN7V 44565798 IC50 = 2 nM T11388 CTHG52 44565799 IC50 = 340 nM T11388 CU9Q2V 44565800 IC50 = 60 nM T11388 CS6MQ7 44565818 IC50 = 22 nM T11388 CM5K6W 44565819 IC50 = 24 nM T11388 CD20NZ 44565820 IC50 = 9 nM T11388 C27FBG 44565821 IC50 = 14 nM T11388 CVO5I7 44565822 IC50 = 32 nM T11388 CA3E8I 44565823 IC50 = 62 nM T11388 C1BH5L 44567669 IC50 = 0.015 nM T11388 CHZ74X 44567681 IC50 = 5 nM T11388 CI6H7R 44568190 IC50 > 2000 nM T11388 CVX81T 44568191 IC50 > 5000 nM T11388 CJRQ74 44568192 IC50 = 390 nM T11388 C6ZHA4 44568193 IC50 = 280 nM T11388 C2X3HJ 44568223 IC50 > 1000 nM T11388 CV54EU 44568306 IC50 > 1500 nM T11388 CDZ03Q 44568307 IC50 > 1000 nM T11388 C6FV7W 44568638 IC50 = 100 nM T11388 C6U3RB 44568639 IC50 = 6 nM T11388 COJ16S 44568640 IC50 = 220 nM T11388 CVP4Y6 44568641 IC50 > 1000 nM T11388 CZW5K2 44568669 IC50 = 17 nM T11388 CW89JM 44568670 IC50 > 1000 nM T11388 C2D9TS 44568671 IC50 > 1000 nM T11388 CU4PO0 44568672 IC50 = 100 nM T11388 CCJ68F 44568673 IC50 > 1000 nM T11388 CCIP49 44568714 IC50 > 1000 nM T11388 C3HYW8 44568715 IC50 > 1000 nM T11388 CLXN21 44568716 IC50 = 280 nM T11388 CU82VX 44568766 IC50 > 1000 nM T11388 CZF5G0 44568767 IC50 > 1000 nM T11388 CVR02S 44568768 IC50 > 1000 nM T11388 C1P3LN 44568769 IC50 = 250 nM T11388 CG74ZL 44568770 IC50 = 480 nM T11388 COHB20 44570671 Ki = 440 nM T11388 C35ZYP 44570672 Ki = 950 nM T11388 C3BHM4 44570673 Ki = 300 nM T11388 C0OSY2 44570674 Ki = 430 nM T11388 CF41YI 44570719 Ki = 1700 nM T11388 CY9ZT4 44570833 Ki = 560 nM T11388 CB3S2D 44570834 Ki = 5000 nM T11388 C8K6PB 44570835 Ki = 240 nM T11388 CWH9Q0 44570836 Ki = 1900 nM T11388 CA10KC 44570876 Ki = 840 nM T11388 CAUD26 44570877 Ki = 700 nM T11388 C1XCP6 44570878 Ki = 750 nM T11388 CN1GT2 44570879 Ki = 730 nM T11388 CV0KJ4 44570915 Ki = 1600 nM T11388 C14JNH 44570916 Ki = 2200 nM T11388 C1DA8K 44570917 Ki = 1200 nM T11388 C9CMZ2 44570957 Ki = 370 nM T11388 C37LRT 44570958 Ki = 520 nM T11388 C31BXW 44570959 Ki = 980 nM T11388 C5G2KT 44570997 Ki = 550 nM T11388 CZ1ET3 44570998 Ki = 950 nM T11388 CSYI14 44570999 Ki = 500 nM T11388 CK5ZM6 44571085 Ki = 950 nM T11388 CNP2G3 44571086 Ki = 730 nM T11388 CX2B3F 44571130 Ki = 820 nM T11388 CFTE86 44571131 Ki = 1100 nM T11388 C4DV1E 44571132 Ki = 570 nM T11388 C05LYD 44571173 Ki = 450 nM T11388 CC5A6D 44571174 Ki = 260 nM T11388 CHB7Y3 44571175 Ki = 800 nM T11388 C6XF8B 44571212 Ki = 1000 nM T11388 CG5ZO3 44571213 Ki = 640 nM T11388 C67UMF 44571214 Ki = 3000 nM T11388 CD6X2Y 44571254 Ki = 1700 nM T11388 CQ0W5J 44571255 Ki = 2300 nM T11388 C6B3IU 44571273 IC50 = 5.7 nM T11388 C4XG6A 44571274 IC50 = 27 nM T11388 C90ORU 44571275 IC50 = 9.8 nM T11388 CGM30J 44571297 Ki = 318 nM T11388 CU0D3P 44571298 Ki = 290 nM T11388 CUG72S 44571323 Ki = 1500 nM T11388 C2NT4H 44571324 Ki = 98 nM T11388 CC12QS 44571325 Ki = 420 nM T11388 CI39YN 44571326 Ki = 23000 nM T11388 CLH46N 44571339 IC50 = 45 nM T11388 CCK6Z3 44571340 IC50 = 0.16 nM T11388 C1L3KX 44571358 Ki = 470 nM T11388 C0NFJ8 44571359 Ki = 1500 nM T11388 CE2PQ4 44571360 Ki = 1200 nM T11388 C5S6FJ 44571361 Ki = 500 nM T11388 C2AVQ0 44587440 IC50 = 240 nM T11388 CO7TR5 44587827 IC50 = 15 nM T11388 CL18MT 44587828 IC50 = 36 nM T11388 C3A4JO 44587829 IC50 = 9 nM T11388 C9HES8 44587858 IC50 = 130 nM T11388 CA4DK2 44587859 IC50 > 3000 nM T11388 C76PSY 44587860 IC50 > 3000 nM T11388 C6NU0J 44587861 IC50 > 1000 nM T11388 CERA06 44587897 IC50 = 200 nM T11388 CNM2G4 44587937 IC50 = 170 nM T11388 CD05MG 46216820 IC50 = 0.4 nM T11388 C4YAJ7 46228924 IC50 > 10000 nM T11388 C6YCT4 46231379 IC50 = 0.4 nM T11388 CQE7G5 46231380 IC50 = 0.3 nM T11388 CVY2P5 46231381 IC50 = 0.5 nM T11388 C8AE2C 46231427 IC50 = 0.2 nM T11388 CLYF89 46231428 IC50 = 0.3 nM T11388 CW1LI8 46231429 IC50 = 0.2 nM T11388 CS1Y5Z 46232305 IC50 = 2.6 nM T11388 C5QE7P 46238539 IC50 = 1660 nM T11388 C1H2RA 46500558 IC50 = 18100 nM T11388 CC2N0F 46842579 IC50 = 708 nM T11388 CV6SW4 46842581 IC50 = 288 nM T11388 CM2D1G 46842582 IC50 = 407 nM T11388 CIU1R5 46842626 IC50 = 1148 nM T11388 C37OSC 46842709 IC50 = 813 nM T11388 C6HD4M 46865101 IC50 = 17 nM T11388 CC7DG3 46866398 IC50 = 10 nM T11388 C38HWY 46878211 Ki = 5.5 nM T11388 CZ43KH 46878212 Ki = 40.1 nM T11388 C4ER8Q 46881086 IC50 = 20.89 nM T11388 C8HX3E 46881090 IC50 = 3.02 nM T11388 C6VA2I 46881091 IC50 = 28.84 nM T11388 CNM34R 46881131 IC50 = 26.92 nM T11388 CVR6J1 46881132 IC50 = 1.585 nM T11388 CJ3H5Z 46881202 IC50 = 1.698 nM T11388 CX1R9T 46881203 IC50 = 6.918 nM T11388 C2LA0F 46881204 IC50 = 57.54 nM T11388 CN04VB 46881205 IC50 = 5.012 nM T11388 C2HOX0 46881206 IC50 = 2.089 nM T11388 CR03YN 46881207 IC50 = 8.913 nM T11388 C12MGB 46881208 IC50 = 14.13 nM T11388 CCQF36 46881221 IC50 = 0.4169 nM T11388 C80DJP 46881268 IC50 = 64.57 nM T11388 C47TYV 46881276 IC50 = 32.36 nM T11388 C4YOJ5 46881277 IC50 = 2.818 nM T11388 C2RHK4 46881278 IC50 = 15.14 nM T11388 C65YCU 46881400 IC50 = 182 nM T11388 C3P5RK 46881401 IC50 = 810 nM T11388 C3Q8KR 46881402 IC50 = 112 nM T11388 CV0I7L 46881403 IC50 = 110 nM T11388 CGT1Z2 46881448 IC50 = 11 nM T11388 CH9ON3 46881449 IC50 = 457 nM T11388 CF15KQ 46881450 IC50 = 148 nM T11388 CJ0XH5 46881452 IC50 = 293 nM T11388 C6O2JN 46881453 IC50 = 96 nM T11388 C9ZXM0 46881456 IC50 = 100 nM T11388 CC78RN 46881457 IC50 = 500 nM T11388 CM3O1Y 46881458 IC50 = 38 nM T11388 CZD09J 46881913 IC50 > 10000 nM T11388 C9Z4OX 46881948 IC50 = 3500 nM T11388 CW3O4C 46881949 IC50 = 72 nM T11388 CHB0Y3 46881950 IC50 = 288 nM T11388 CN59JW 46881951 IC50 > 10000 nM T11388 C8SJ2P 46881952 IC50 > 10000 nM T11388 CUVD91 46881953 IC50 > 10000 nM T11388 C4W5CQ 46881995 IC50 = 870 nM T11388 CLP21F 46881996 IC50 = 197 nM T11388 C9E4RV 46881997 IC50 = 38 nM T11388 C2XLY3 46881998 IC50 = 1100 nM T11388 C4VN0T 46881999 IC50 = 7400 nM T11388 C4S9CR 46882040 IC50 = 2000 nM T11388 CT8EW1 46882041 IC50 = 12000 nM T11388 CW10YO 46882042 IC50 = 1000 nM T11388 CHIV65 46882043 IC50 = 4460 nM T11388 CMJC43 46882044 IC50 = 100 nM T11388 CN58BG 46882092 IC50 = 33 nM T11388 CG9X3C 46882094 IC50 = 4070 nM T11388 CZ5KP8 46882095 IC50 = 977 nM T11388 CPQZ83 46882096 IC50 = 34 nM T11388 CHX21M 46882097 IC50 = 1000 nM T11388 CA30PF 46889752 Ki = 2.5 nM T11388 C50BXV 46911628 IC50 = 3090 nM T11388 CYG6M1 46911633 IC50 = 1072 nM T11388 CTW1Q2 46911634 IC50 = 2291 nM T11388 C07GBO 46911635 IC50 = 117 nM T11388 CFWU08 46946224 IC50 > 25000 nM T11388 CVT40A 46947220 IC50 > 25000 nM T11388 CAFW31 49783666 IC50 > 10000 nM T11388 CGF65B 49783985 IC50 = 7943.28 nM T11388 C4NB3R 49834903 IC50 > 25000 nM T11388 CQ3W9J 49834904 IC50 > 25000 nM T11388 CX1WU8 49834905 IC50 > 25000 nM T11388 CA96LF 49834906 IC50 > 25000 nM T11388 CB9MS2 49834907 IC50 > 25000 nM T11388 C74RAF 49834908 IC50 > 25000 nM T11388 CN8E2A 49834971 IC50 > 25000 nM T11388 COG9T6 49834972 IC50 > 25000 nM T11388 CGPM91 49834975 IC50 > 25000 nM T11388 CJ73DH 49835032 IC50 > 25000 nM T11388 C8XR4Q 49835033 IC50 > 25000 nM T11388 CXE51M 49835035 IC50 > 25000 nM T11388 CKRG17 49835144 IC50 > 25000 nM T11388 C9NO4U 49835145 IC50 > 25000 nM T11388 CS23QM 49835147 IC50 > 25000 nM T11388 CCO0S5 49835202 IC50 > 25000 nM T11388 CP4S5A 49835673 IC50 = 15500 nM T11388 CS3HC6 49835674 IC50 = 29700 nM T11388 CSTC36 49835675 IC50 > 25000 nM T11388 C8O3UF 49835732 IC50 > 25000 nM T11388 CU56CD 49862015 IC50 > 10000 nM T11388 CMA62P 49862016 IC50 > 10000 nM T11388 COY8Z0 49862017 IC50 > 10000 nM T11388 CEH26G 49862059 IC50 = 1259 nM T11388 CEHY57 49862060 IC50 = 3162 nM T11388 CI90VX 49862061 IC50 = 1071 nM T11388 C6QN8X 49862100 IC50 > 10000 nM T11388 CFB57Z 49862101 IC50 > 10000 nM T11388 CCM26G 49862102 IC50 = 2042 nM T11388 CDZL08 49862143 IC50 = 2512 nM T11388 CVB95I 49862144 IC50 = 891 nM T11388 CWG62C 49862145 IC50 = 240 nM T11388 C37RZT 49862146 IC50 = 178 nM T11388 CGT50H 49862184 IC50 = 5888 nM T11388 CO1Y6B 49862185 IC50 = 1175 nM T11388 CJ0HY8 49862186 IC50 = 776 nM T11388 CD97QU 49862228 IC50 = 13 nM T11388 CXO39G 49862275 IC50 > 10000 nM T11388 CKA53W 49862308 IC50 = 60 nM T11388 C8B2WE 49862309 IC50 = 44 nM T11388 CR13LF 49862310 IC50 = 316 nM T11388 C38BJK 49862365 IC50 = 71 nM T11388 C1Z9VQ 49862366 IC50 = 166 nM T11388 C6W1UJ 49862367 IC50 = 56 nM T11388 CIFP19 49862368 IC50 = 398 nM T11388 CMW23V 49862369 IC50 = 661 nM T11388 CI4J0A 49862370 IC50 = 195 nM T11388 C1XBM6 49862420 IC50 = 145 nM T11388 CKV06S 49862421 IC50 = 44 nM T11388 CN4GD6 49862422 IC50 = 1000 nM T11388 CA7K8Q 49862423 IC50 = 32 nM T11388 CS92IZ 49862471 IC50 = 17 nM T11388 C1NAQ5 49862472 IC50 = 151 nM T11388 C5OD6J 49862473 IC50 = 40 nM T11388 CFCH31 49862474 IC50 = 65 nM T11388 C29OGE 49862475 IC50 = 91 nM T11388 CU7T1N 49862476 IC50 = 470 nM T11388 CW36FO 49862535 IC50 = 630 nM T11388 CM94UQ 49862536 IC50 = 282 nM T11388 C69TUQ 49862719 IC50 > 10000 nM T11388 CTQ19U 49862720 IC50 > 10000 nM T11388 CN6L9Y 49862793 IC50 = 1995 nM T11388 CN8PD3 49862794 IC50 = 8511 nM T11388 CU3QE7 49862795 IC50 = 2818 nM T11388 COA12C 49862796 IC50 = 7762 nM T11388 C3N8YJ 49862797 IC50 = 2691 nM T11388 CZPY13 49863204 IC50 = 50 nM T11388 C5GU2F 49863239 IC50 = 8900 nM T11388 CN9PI1 49867423 IC50 < 1 nM T11388 C18RNG 50925386 Ki = 0.63 nM T11388 C01DJG 50993971 Ki = 260 nM T11388 CW9X3R 50993972 Ki = 33 nM T11388 CIC7H1 50993973 Ki = 0.87 nM T11388 C3UB9Y 50993974 Ki = 0.46 nM T11388 CMS13V 50994055 Ki = 0.071 nM T11388 CPT6I5 50994056 Ki = 0.16 nM T11388 CB4X6Y 50994057 Ki = 0.017 nM T11388 CSY4W0 50994058 Ki = 0.011 nM T11388 CQ08HC 50994059 Ki = 0.11 nM T11388 C30WKN 50994060 Ki = 0.072 nM T11388 C8A1GN 50994137 Ki = 0.045 nM T11388 C6K3EJ 50994138 Ki = 0.022 nM T11388 CN6ZM0 50994139 Ki = 34 nM T11388 CF7SN9 50994140 Ki = 2.9 nM T11388 CU7M1P 50994141 Ki = 270 nM T11388 C4FE0T 50994142 Ki = 0.032 nM T11388 CZP0H6 51003522 IC50 = 0.8 nM T11388 CH5S0P 52940936 IC50 = 5 nM T11388 CKP92N 52941058 IC50 = 30 nM T11388 CDC64G 52941172 IC50 > 10000 nM T11388 CJSD25 52941466 IC50 = 51.3 nM T11388 C71VFU 52941469 IC50 = 11.7 nM T11388 CBKG58 52941965 IC50 > 10000 nM T11388 C51MIQ 52942095 IC50 = 4 nM T11388 C3E5WI 52942171 IC50 = 4 nM T11388 CL65FB 52942200 IC50 = 10 nM T11388 C3WH6F 52942248 IC50 = 9 nM T11388 CFP83K 52942699 IC50 = 26.3 nM T11388 CBM6K7 52942707 IC50 = 33.1 nM T11388 C12MHY 52942758 IC50 = 91.2 nM T11388 CW05MV 52942797 IC50 = 20.9 nM T11388 C8IC1X 52943191 IC50 > 10000 nM T11388 CNI79L 52943227 IC50 = 9 nM T11388 CJWI80 52943409 IC50 = 11 nM T11388 CQDG96 52943578 IC50 = 46.8 nM T11388 C25NCO 52944522 IC50 = 8 nM T11388 CO85FM 52944637 IC50 = 3 nM T11388 C9RY6V 52945164 IC50 = 195 nM T11388 CL1RH9 52945722 IC50 = 427 nM T11388 C1Z9HY 52945786 IC50 = 13 nM T11388 CF46DK 52945849 IC50 = 9 nM T11388 C9B1ON 52946392 IC50 = 37.2 nM T11388 C5CJT3 52946393 IC50 = 8.7 nM T11388 C2GVW6 52947078 IC50 = 9 nM T11388 CD6CT7 52948442 IC50 = 11.5 nM T11388 CTV1C2 52948769 IC50 = 107.2 nM T11388 C75SHQ 52948860 IC50 = 12.9 nM T11388 CLIS74 52948911 IC50 = 32 nM T11388 C25FAX 52948924 IC50 = 389 nM T11388 C9YWD1 52949393 IC50 = 12 nM T11388 CROV43 52949411 IC50 = 166 nM T11388 C0AZH4 52949420 IC50 = 6 nM T11388 CRL18H 52949508 IC50 = 12 nM T11388 C3TB7W 52949669 IC50 = 47.9 nM T11388 C56OCA 53317528 IC50 = 1258.93 nM T11388 C7I9AO 53317529 IC50 = 10000 nM T11388 CM60RJ 53317530 IC50 = 5011.87 nM T11388 C6FEH9 53318816 IC50 > 25118.86 nM T11388 CJAX07 53318817 IC50 = 1000 nM T11388 CG5AP6 53318818 IC50 = 630.96 nM T11388 C2Z1XT 53318875 IC50 = 1.9 nM T11388 CBM79Y 53320190 IC50 = 0.3 nM T11388 C7V2DA 53322116 IC50 = 1905 nM T11388 CQ8O1R 53322117 IC50 = 2344 nM T11388 C0QV5D 53322753 IC50 = 63.1 nM T11388 CH8Q6D 53322840 IC50 = 0.3 nM T11388 CZWL65 53324168 IC50 = 1.6 nM T11388 CHB96K 53324300 IC50 = 199.53 nM T11388 CR1L4Y 53325394 IC50 > 25118.86 nM T11388 CVU0J1 53326656 IC50 = 31.62 nM T11388 CWJB05 53364091 IC50 = 263 nM T11388 CA01ZV 54704806 IC50 = 4600 nM T11388 CCG3S4 56666730 IC50 = 10 nM T11388 CK54CF 56670150 IC50 = 1 nM T11388 C69ILG 56670151 IC50 = 11.2 nM T11388 CA2Z0U 56676986 IC50 = 6200 nM T11388 C24QMN 56680316 IC50 = 1900 nM T11388 CX8M7Z 56683636 IC50 = 27.7 nM T11388 C84CHB 57541268 IC50 = 1 nM T11388 CH72FA 57541295 IC50 = 25 nM T11388 C6J3FL 59028747 IC50 = 81 nM T11388 CH3M0B 59543520 IC50 > 25000 nM T11388 CCR9Q8 59543629 IC50 > 25000 nM T11388 C3ESJ1 59543757 IC50 > 25000 nM T11388 CZV45P 59619390 IC50 > 25000 nM T11388 CLX2Y4 60148518 Ki > 40000 nM T11388 C0DA6M 60166364 Ki > 40000 nM T11388 C4G1SF 60166365 Ki > 40000 nM T11388 COM7U3 60166366 Ki > 4000 nM T11388 COQ82A 60166367 Ki > 4000 nM T11388 C2Y7EK 60166492 Ki > 4000 nM T11388 C4PHR1 60166493 Ki > 4000 nM T11388 CG4DZ7 60166494 Ki > 4000 nM T11388 C5E2PB 60166495 Ki = 1100 nM T11388 CXD39V 60166496 Ki > 4000 nM T11388 CM8XO5 60166497 Ki > 4000 nM T11388 CA95CZ 60195809 IC50 = 257 nM T11388 CY3VC4 60195810 IC50 = 73 nM T11388 CMA8T3 60195811 IC50 = 18 nM T11388 CVRJ91 60195812 IC50 = 2 nM T11388 CE6AH0 60195813 IC50 = 37 nM T11388 C8ILH6 60195902 IC50 = 7 nM T11388 CX4N2V 60195903 IC50 < 1 nM T11388 C4PQ6E 60195904 IC50 = 16.2 nM T11388 CNUI89 60195905 IC50 = 17.3 nM T11388 C23JUZ 60195906 IC50 = 785 nM T11388 CSF35K 70274227 IC50 = 12 nM T11388 CI0XF8 70274815 IC50 = 19.95 nM T11388 CXT5G7 70275845 IC50 = 59 nM T11388 C5P3BO 70275923 IC50 = 211 nM T11388 C3U9IH 70276243 IC50 = 199.53 nM T11388 CCG16F 70276365 IC50 = 31.62 nM T11388 C0T3LC 70276605 IC50 = 9 nM T11388 CE1J0O 70276811 IC50 = 25.12 nM T11388 C06WFN 70276830 IC50 = 316.23 nM T11388 CDQ85E 70276990 IC50 = 25.12 nM T11388 CGET13 70278898 IC50 = 15 nM T11388 C2GT5H 70280758 IC50 = 25.12 nM T11388 CI53XU 70281040 IC50 = 45 nM T11388 CA6DM2 70281073 IC50 = 25.12 nM T11388 CE70MT 70676095 IC50 = 12470 nM T11388 CS8VR4 70676096 IC50 = 5720 nM T11388 CZ84UX 70682584 IC50 = 31.62 nM T11388 CL9RE3 70686820 IC50 = 19.95 nM T11388 C65EDY 70686822 IC50 = 12.59 nM T11388 C5IYR0 70688897 IC50 = 19.95 nM T11388 CZOF81 70693115 IC50 = 10 nM T11388 CMFW03 70693116 IC50 = 63.1 nM T11388 C5RSJ0 70693117 IC50 = 15.85 nM T11388 C01IDC 70695171 IC50 = 15.85 nM T11388 CO4J7W 70695553 IC50 = 200 nM T11388 CURI37 70696209 Ki = 5.75 nM T11388 C34WHG 70697225 IC50 = 39.81 nM T11388 CUB38S 71449749 IC50 = 3 nM T11388 C08LGJ 71451733 IC50 = 23 nM T11388 CI7Z8B 71451734 IC50 = 9 nM T11388 C7RJG8 71453558 IC50 = 11 nM T11388 C2OGP1 71453559 IC50 = 25 nM T11388 CDR10X 71453560 IC50 = 15 nM T11388 CPGT63 71454020 Ki = 230 nM T11388 CFUS41 71455276 IC50 = 11 nM T11388 CUQL74 71455277 IC50 = 17 nM T11388 C0KUW5 71455278 IC50 = 5 nM T11388 C7Z0HF 71455279 IC50 = 11 nM T11388 CU48QH 71455759 Ki = 880 nM T11388 C9YJG7 71457065 IC50 = 6 nM T11388 CCH47M 71458921 IC50 = 14 nM T11388 CP7MZ5 71458922 IC50 = 9 nM T11388 CCA46N 71458923 IC50 = 4 nM T11388 CQT1C2 71458924 IC50 = 6 nM T11388 C6RZF3 71459429 Ki = 19 nM T11388 CE9LP1 71460574 IC50 = 3 nM T11388 CDW0I7 71460731 IC50 = 6 nM T11388 CC87WL 71460732 IC50 = 8 nM T11388 CL6Y4C 71460733 IC50 = 16 nM T11388 CER82H 71612695 Ki = 24000 nM T11388 C5NV8E 71624115 IC50 > 10000 nM T11388 C8DZ6U 71624118 IC50 > 10000 nM T11388 C8SGK6 71624246 IC50 > 10000 nM T11388 CM64QD 71624362 IC50 > 10000 nM T11388 CK64NT 71624363 IC50 > 10000 nM T11388 CAN6X5 71656574 IC50 >= 25000 nM T11388 CB8EY9 71716783 IC50 = 0.83 nM T11388 CDP94C 71717397 Ki = 11.5 nM T11388 C71AQG 71717398 IC50 = 19600 nM T11388 CSN07F 72793721 IC50 > 25000 nM T11388 C6I4RC 72793722 IC50 > 25000 nM T11388 CO1W8E 72793723 IC50 > 25000 nM T11388 CY1IU2 73345852 Ki = 639000 nM T11388 C0HSC8 73346520 Ki = 23950 nM T11388 C8SD9P 73346521 Ki = 49780 nM T11388 CGZ6Y8 73346522 Ki = 44900 nM T11388 C43IPQ 73348006 Ki = 4580 nM T11388 CJQE58 73348851 Ki = 47000 nM T11388 C31JUR 73348857 Ki = 147000 nM T11388 C95BEA 73348858 Ki = 284000 nM T11388 CS9C0W 73351108 Ki = 8710 nM T11388 CAYM96 73351955 Ki = 213000 nM T11388 C27JUH 73352576 Ki = 24150 nM T11388 CVP03Z 73352577 Ki = 6220 nM T11388 CDAB86 73354065 Ki = 10770 nM T11388 CK3Z8U 73354066 Ki = 11610 nM T11388 C92DXZ 73354067 Ki = 51240 nM T11388 CCI18Y 73355591 Ki = 11120 nM T11388 CRX8A0 73355592 Ki = 21870 nM T11388 CJ6CQ1 73356205 Ki = 77 nM T11388 C0ZDB4 76313697 IC50 = 16 nM T11388 CX26GW 76328142 IC50 = 855 nM T11388 C62SML 90655967 IC50 = 251.19 nM T11388 CJ7LT3 90655968 IC50 = 6309.57 nM T11388 CB61WC 90655969 IC50 = 7943.28 nM T11388 CIS56R 90663177 Ki = 230 nM T11388 CU71EO 90663180 Ki = 30500 nM T11388 CJ2V9B 90663412 Ki = 2900 nM T11388 C89DWE 90663417 Ki = 1000 nM T11388 CX9I6Z 90663418 Ki = 5900 nM T11388 C0XZH3 90665919 IC50 = 14520 nM T11388 C0HIA4 90665921 IC50 = 5620 nM T11388 CH68BZ 91885514 Ki = 22 nM T11388 CRVO29 91885636 Ki = 10 nM T11388 CTE34I 118720232 IC50 > 100000 nM T11388 CSD62B 118720233 IC50 > 100000 nM T11388 C9WF7Q 118720234 IC50 = 9500 nM T11388 C76HIO 118720235 IC50 = 19000 nM T11388 CAT1R6 118720236 IC50 > 100000 nM T11388 CGAF42 118720237 IC50 = 95000 nM T11388 CJ28KZ 118720238 IC50 = 73000 nM T11388 CPH2V9 118720239 IC50 > 100000 nM T11388 CCXD81 122186478 Ki = 70 nM T11388 C35TQG 122186479 Ki = 16 nM T11388 CF0CG5 122186480 Ki > 500 nM T11388 CIP70Z 122186481 Ki = 114 nM T11388 C3C7BJ 122186482 Ki = 55 nM T11388 CIG4L8 122197311 IC50 = 9600 nM T11388 CMT2B9 127049869 Ki = 370 nM T11388 C43APM 127050163 Ki = 580 nM T11388 C8VKA5 127050164 Ki = 370 nM T11388 CZ54XC 127050165 Ki = 67.6 nM T11388 CI2C3V 127050166 Ki = 335 nM T11388 C7V8XZ 127051317 Ki = 226 nM T11388 CSK16Q 127051318 Ki = 535 nM T11388 C7YI4M 127051342 Ki = 4500 nM T11388 C6NFU9 127051343 Ki = 930 nM T11388 C6SD7P 127051344 Ki = 24.5 nM T11388 CY5CV6 127051345 Ki = 310 nM T11388 C6DCO9 132937452 Ki = 11 nM T11388 C2CT4O 134134083 IC50 = 68 nM T11388 C89UGK 134134373 Ki = 41 nM T11388 CX7UT0 134135239 IC50 = 70 nM T11388 COU6A4 134135795 IC50 = 28 nM T11388 CD0UE9 134136855 IC50 = 17 nM T11388 CF8VA4 134138144 IC50 = 17 nM T11388 CFE54U 134139713 IC50 = 60 nM T11388 CQ8U5W 134141808 IC50 = 28 nM T11388 C3PEW2 134141970 IC50 = 17 nM T11388 CV36BU 134142724 IC50 = 23 nM T11388 C4BXO1 134144535 IC50 = 17 nM T11388 C9I7CY 134146605 Ki = 393 nM T11388 CE8Q2J 134147121 IC50 = 80 nM T11388 C8WYF6 134147241 IC50 = 34 nM T11388 C0YG8C 134148335 IC50 = 23 nM T11388 C7CH0G 134151560 IC50 = 67 nM T11388 CELG81 134154408 Ki = 163 nM T11388 C4TS3J 134154893 IC50 = 17 nM T11388 CP1B6I 135533094 IC50 = 3400 nM T11388 CM54ID 137655962 Ki = 44000 nM T11388 CFQ25D 145967499 IC50 = 867 nM T11388 CIVB10 145967715 IC50 = 1 nM T11388 CLI6T0 145967952 IC50 > 5000 nM T11388 CC4AG7 145968405 IC50 > 5000 nM T11388 CDS31M 145968622 IC50 = 1.3 nM T11388 CA40YU 145969275 IC50 = 213 nM T11388 CB0Y7Z 145969438 IC50 = 3828 nM T11388 C2WCK0 145969450 IC50 = 2690 nM T11388 CL7KO9 145969878 IC50 = 435 nM T11388 C3NAS7 145970030 IC50 > 5000 nM T11388 CS08XI 145970918 IC50 > 5000 nM T11388 C9XKW2 145970931 IC50 = 1870 nM T11388 CQ3TG0 145979639 Ki = 800 nM T11388 CXW3F1 145982578 IC50 = 100 nM T11388 CY7XE4 145982644 IC50 = 400 nM T11388 C56AXR 145982654 IC50 = 30 nM T11388 C7S2TX 145983004 IC50 = 60 nM T11388 C7V2ZF 145983823 IC50 = 50 nM T11388 CV1A6D 145983891 Ki = 700 nM T11388 CV8HP6 145984203 Ki = 3 nM T11388 C3JIQ4 145984217 IC50 = 500 nM T11388 CT8QM9 145984597 IC50 = 800 nM T11388 CJM6L4 145984752 IC50 = 20 nM T11388 C0BC2Z 145984777 IC50 = 100 nM T11388 CGC54P 145985016 IC50 = 100 nM T11388 C2LB8K 145985094 IC50 = 100 nM T11388 CNT63X 145985191 IC50 = 30 nM T11388 CX6JT1 145985564 IC50 = 200 nM T11388 CJE7L9 145985615 IC50 = 700 nM T11388 CL2B3Y 145985677 IC50 = 600 nM T11388 CQ2RS8 145986120 IC50 = 200 nM T11388 CM53FT 145986712 Ki = 3 nM T11388 C6OKB9 145987263 IC50 > 5000 nM T11388 CRD65W 145987430 Ki = 10000 nM T11388 COZ6P5 145987960 IC50 > 5000 nM T11388 C7ZCW3 145988622 IC50 > 5000 nM T11388 C9OAK6 145989037 IC50 = 0.11 nM T11388 C87GKT 145989707 IC50 = 202 nM T11388 C5MWT1 145990477 Ki = 9 nM T11388 CBN12I 155524050 Ki = 7.21 nM T11388 CXYT09 155551122 Ki = 1.14 nM T11388 CHD79T 44408017 IC50 = 48 nM T11388 CO0N3S 44408050 IC50 = 1.1 nM T11388 CY4JN6 44408058 IC50 = 59 nM T11388 CN8Y0L 44408080 IC50 = 110 nM T11388 C58OLD 44517711 IC50 = 1000 nM T11388 CT3S1I 44517712 IC50 = 158.49 nM T11388 CFT38D 45267632 IC50 = 6309.57 nM T11388 COU83P 45267640 IC50 = 630.96 nM T11388 C1U4IF 45267645 IC50 = 3162.28 nM T11388 CDG5S8 45268499 IC50 > 10000 nM T11388 CV8PZ3 45268510 IC50 > 10000 nM T11388 C89ADF 45269361 IC50 > 10000 nM T11388 C58PZI 45269375 IC50 = 1258.93 nM T11388 C5O9EF 45270206 IC50 = 125.89 nM T11388 C07ADH 45270207 IC50 = 125.89 nM T11388 CVGE81 45270212 IC50 = 100 nM T11388 C78EXG 45271021 IC50 > 7943.28 nM T11388 C5MBC4 45271038 IC50 = 63.1 nM T11388 C65QLD 45271887 IC50 > 7943.28 nM T11388 CIL8O6 45271888 IC50 > 10000 nM T11388 CLFD35 45272742 IC50 > 10000 nM T11388 C3WF8S 45272748 IC50 > 10000 nM T11388 CQO98K 45272752 IC50 > 6309.57 nM T11388 C9A0IH 45272753 IC50 = 125.89 nM T11388 CSYU09 45273681 IC50 > 10000 nM T11388 D00FGA 73737 IC50 = 1000 nM T11388 D00QIA 104275 IC50 = 31 nM T11388 D00TRY 448022 IC50 = 26 nM T11388 D01IFO 49863205 IC50 > 10000 nM T11388 D01JGB 46881498 IC50 = 11 nM T11388 D01YNC 23648531 Ki = 5800 nM T11388 D02TNR 17945750 IC50 = 78 nM T11388 D04BGT 46881451 IC50 = 182 nM T11388 D04QHB 16108885 IC50 = 120 nM T11388 D05WZF 10129151 IC50 = 40 nM T11388 D06AZJ 16108884 IC50 = 170 nM T11388 D06VIP 14774521 Ki = 6500 nM T11388 D06WQP 60148519 Ki = 0.66 nM T11388 D07FLB 11637576 Ki = 1270 nM T11388 D07RSA 11696652 Ki = 300 nM T11388 D07SOQ 11652399 Ki > 100000 nM T11388 D08KCA 72429 IC50 = 0.018 ug.mL-1 T11388 D09AHN 11492732 Ki = 120 nM T11388 D09FGQ 123985 IC50 = 4 nM T11388 D0A7ER 11514386 Ki = 1100 nM T11388 D0A8OV 11086036 Ki = 7500 nM T11388 D0B2FE 46882093 IC50 = 1122 nM T11388 D0D0LD 9913088 IC50 = 0.2 nM T11388 D0FC7L 16108897 IC50 = 1000 nM T11388 D0G2QG 44343301 IC50 = 1.8 nM T11388 D0G8OD 11702208 Ki = 35 nM T11388 D0H8CC 44398742 Ki = 60 nM T11388 D0JF8D 11551481 Ki = 30000 nM T11388 D0JN8Q 11702265 Ki = 1500 nM T11388 D0L9VP 5287864 Ki = 1.2 nM T11388 D0P5BY 11550059 IC50 = 3400 nM T11388 D0Q4UA 10033311 Ki = 21 nM T11388 D0T7QF 10420833 IC50 = 51 nM T11388 D0U0XG 11709032 Ki = 730 nM T11388 D0U4TY 11694425 IC50 = 84 nM T11388 D0VE0F 10062714 IC50 = 0.35 nM T11388 D0Y5IQ 44255320 IC50 = 10000 nM T11388 D0Y5LX 11622731 IC50 = 680 nM T11388 D0Z0PR 9912381 IC50 = 0.25 nM T77063 CUS16Z 44584846 Ki = 562 nM T77063 CP2J8X 44584953 Ki = 515 nM T77063 CBX8K0 44584960 Ki = 952 nM T77063 C10KCB 44584961 Ki = 772 nM T77063 C1S6KQ 44584962 Ki = 624 nM T77063 D05JJL 44584947 Ki = 441 nM T01396 D0E3TC 44259 IC50 = 0.133 nM T01396 D0T3ME 156422 IC50 = 43000 nM T01396 CBOP58 11293798 Ki > 10000 nM T01396 C26BZX 11362471 Ki = 7350 nM T01396 CWXB93 11397177 Ki > 10000 nM T01396 CTG83F 11539329 Ki > 7500 nM T01396 CMIL86 11590363 Ki > 7500 nM T01396 C9T6SC 11640926 Ki > 7500 nM T01396 CFPW41 16007116 Ki > 7500 nM T01396 CETQ79 44427518 IC50 = 13860 nM T01396 COPG94 44427519 IC50 > 10000 nM T01396 C3VRO9 44557921 IC50 > 10000 nM T01396 C8NA4L 53384644 IC50 > 30000 nM T01396 C1MR8Q 60097495 IC50 > 1000 nM T01396 CV63UL 67240318 IC50 > 10000 nM T01396 CKT60L 71455860 Ki = 3610 nM T01396 CRJ45X 135589980 IC50 > 50000 nM T01396 C26ESH 136060555 IC50 = 4590 nM T01396 C2MD1Q 155513187 IC50 > 10000 nM T01396 D00ERW 44444843 Ki = 4266 nM T01396 D00HVA 11624601 Ki > 7500 nM T01396 D0Q3NG 11715520 Ki > 7500 nM T01396 D0S7IE 11658882 Ki > 7500 nM T45299 D05PHH 3447 IC50 = 15360 nM T45299 D07UWV 92722 Ki = 87800 nM T45299 D0I0RJ 16231 IC50 > 20000 nM T45299 D0J0BU 10275777 IC50 > 10000 nM T45299 D0M7JT 216210 Ki = 45360 nM T45299 D00LOB 9866964 Ki = 2400 nM T45299 D01MUU 183797 Ki = 900 nM T45299 D0I7MX 9871765 Ki = 433 nM T45299 D0ID3W 9911502 IC50 > 25100 nM T45299 D02QTV 122267 IC50 = 34 nM T45299 D0D5RH 11641515 IC50 = 44000 nM T45299 D0S2JG 9913629 Ki = 27200 nM T45299 D0Y5EX 122296 Ki = 5.7 nM T45299 C71WRJ 1503 Ki = 63000 nM T45299 CY5B9C 1504 Ki = 1000 nM T45299 C2KE5Q 1508 Ki = 9400 nM T45299 C4S1PB 4300 Ki = 256000 nM T45299 CL1T7V 4301 Ki = 10000 nM T45299 C0YU1V 16157 Ki = 733000 nM T45299 CMG15V 122129 Ki = 21000 nM T45299 C1BHS3 193409 Ki > 100000 nM T45299 CZP0Y1 204101 Ki > 33000 nM T45299 C2Z0XW 445482 Ki = 360 nM T45299 CR4KE5 445844 Ki = 110 nM T45299 CU6X2A 445847 Ki = 61000 nM T45299 C5UX1L 447478 Ki = 590 nM T45299 CVND42 447482 Ki = 1000 nM T45299 C4OKV5 447486 Ki = 16000 nM T45299 CC9G5O 447490 Ki = 29000 nM T45299 CR2DX3 447496 Ki = 3400 nM T45299 COYS31 447502 Ki = 46000 nM T45299 CVI28M 447508 Ki = 460 nM T45299 CS09BE 447510 Ki = 2400 nM T45299 C87GLP 447540 Ki = 58000 nM T45299 C87OTC 447733 Ki = 58400 nM T45299 CF6D4B 447734 Ki = 3390 nM T45299 CHT05K 447735 Ki = 1840 nM T45299 C5QKC3 448605 Ki = 680 nM T45299 CX5MS1 448610 Ki = 24000 nM T45299 CFO39X 4369278 Ki = 640 nM T45299 C8I0VG 5289529 Ki > 100000 nM T45299 C7SYK9 6102731 IC50 > 33000 nM T45299 C2ZRF5 6540265 Ki > 100000 nM T45299 CN57IY 6540268 Ki > 100000 nM T45299 CX34ZD 9549214 Ki > 1800 nM T45299 C6JDM9 9799627 Ki = 1650 nM T45299 CKA6C4 9802514 Ki > 100000 nM T45299 C4VX9Y 9803558 IC50 > 10000 nM T45299 C1FIN6 9804775 IC50 > 130 nM T45299 C4OTK6 9805415 IC50 > 10000 nM T45299 CAG59M 9808035 Ki > 10000 nM T45299 CH9IE6 9808346 Ki = 68200 nM T45299 C2AXV0 9809479 Ki > 33000 nM T45299 CKN89B 9822176 Ki = 1900 nM T45299 C1D4EC 9822928 Ki = 38000 nM T45299 CS1DL7 9826716 IC50 = 18000 nM T45299 CGN48U 9827867 IC50 > 2500 nM T45299 C8Z5TX 9843775 Ki > 100000 nM T45299 CS9HQ0 9850467 IC50 = 93 nM T45299 CL6QS0 9868922 Ki = 7400 nM T45299 CDU85Y 9871868 Ki = 24000 nM T45299 C2F5NS 9884570 Ki = 350 nM T45299 CQP0V2 9886960 Ki = 240 nM T45299 C17NPU 9890541 IC50 > 2500 nM T45299 CNJ0W1 9893177 IC50 = 540 nM T45299 CKDP84 9895193 Ki = 4900 nM T45299 CMC95R 9910164 Ki = 106 nM T45299 C13XPD 9912856 Ki > 2500 nM T45299 CC0D5H 9915041 Ki > 33000 nM T45299 C2UX6D 9930716 Ki > 100000 nM T45299 CB7VR2 9934590 IC50 = 6600 nM T45299 CNE25D 9935474 Ki = 34700 nM T45299 C1XT2Y 9935746 Ki > 60000 nM T45299 CL2NV0 9935925 IC50 > 870 nM T45299 CC9QH7 9937406 IC50 = 495 nM T45299 C8F5CW 9937921 Ki > 45000 nM T45299 C8LR4T 9938917 Ki > 33000 nM T45299 CDT95S 9939426 Ki = 2510 nM T45299 C1K5WI 9948854 Ki = 52000 nM T45299 CFK05S 9949275 Ki = 15500 nM T45299 C1RHT8 9949886 Ki = 110 nM T45299 CYP6S7 9952109 Ki = 40000 nM T45299 CW7TZ6 9953704 IC50 > 2500 nM T45299 CD7ZO5 9954791 Ki = 140 nM T45299 C0R4GE 9954812 IC50 = 109000 nM T45299 CX85LD 9954980 Ki > 20000 nM T45299 CM7IF6 9956559 Ki > 20000 nM T45299 CCQE85 9956843 Ki = 34400 nM T45299 CYLI95 9956922 Ki = 23000 nM T45299 C2Y0QV 9959268 IC50 > 10000 nM T45299 CBC2K3 9959749 IC50 > 11000 nM T45299 CZ3U8E 9984568 Ki = 4300 nM T45299 CKIP10 9987251 IC50 = 4600 nM T45299 CVQN23 10003356 Ki = 1400 nM T45299 CFQV59 10007890 IC50 > 10000 nM T45299 C8ME3O 10024183 Ki = 2000 nM T45299 CBL8D4 10026170 Ki = 680 nM T45299 CF1V4K 10027758 Ki > 8700 nM T45299 C4QUM5 10048688 IC50 = 680 nM T45299 C9R8YW 10048823 Ki = 840 nM T45299 CVY28G 10051489 Ki = 110 nM T45299 C3QP6V 10052373 Ki = 3500 nM T45299 CXZ2V3 10054210 Ki = 33000 nM T45299 C6F4SZ 10067786 Ki = 0.29 nM T45299 CF4R2W 10074230 IC50 = 8700 nM T45299 CUOC38 10074752 Ki = 290 nM T45299 CD5AT6 10075317 Ki = 8900 nM T45299 C3TWI1 10095455 Ki > 100000 nM T45299 C3OG5U 10095865 IC50 = 5010 nM T45299 C17CDJ 10096845 IC50 > 2500 nM T45299 CRS8D1 10098302 Ki = 67 nM T45299 CW4RZ5 10116936 IC50 > 450 nM T45299 C1VT4F 10117027 Ki = 67000 nM T45299 C5E0SY 10126451 Ki = 4740 nM T45299 C5VJE7 10131165 Ki = 272000 nM T45299 CS2G4T 10140847 Ki = 8300 nM T45299 C31QAL 10143532 Ki > 33000 nM T45299 C7L5IJ 10157296 Ki = 176 nM T45299 CL7U8P 10181581 Ki = 18943 nM T45299 C7PC2K 10185292 IC50 > 170 nM T45299 CFIH78 10185526 IC50 > 33000 nM T45299 CO51ZR 10205659 IC50 > 10000 nM T45299 CEP79T 10216518 Ki = 4017 nM T45299 C8V1AY 10225952 Ki = 3300 nM T45299 C2XHG8 10248900 Ki = 1700 nM T45299 C4Z1LU 10255253 Ki > 8700 nM T45299 CUX40O 10258264 Ki = 570 nM T45299 CQ9ZO1 10275412 Ki > 43000 nM T45299 C0J1TD 10278414 Ki = 810 nM T45299 CNAX45 10287785 Ki = 7038 nM T45299 C5EDW1 10294146 Ki = 870 nM T45299 CV10CU 10297977 IC50 > 10000 nM T45299 C1AP6H 10298858 IC50 > 10000 nM T45299 C8SQ1N 10324263 Ki > 60000 nM T45299 CX9J5U 10324635 Ki = 100 nM T45299 CP64HV 10342843 Ki > 1000000 nM T45299 CK9J7X 10343728 IC50 > 25100 nM T45299 CF9Q3K 10345602 Ki = 200000 nM T45299 C9XUD8 10347489 IC50 > 33000 nM T45299 C10ISY 10367012 Ki = 137000 nM T45299 CJ0O5P 10367277 IC50 > 33000 nM T45299 CMNP39 10389039 IC50 > 10000 nM T45299 C47OZV 10390121 Ki = 240 nM T45299 C8EPN7 10390481 Ki = 190000 nM T45299 C3BR5A 10390490 Ki = 96 nM T45299 CJNV62 10391699 IC50 > 33000 nM T45299 C6S4CO 10391715 Ki > 60000 nM T45299 CEH4D1 10391881 Ki > 100000 nM T45299 CLK08Z 10391999 IC50 > 10000 nM T45299 C4FBO0 10409093 Ki = 2900 nM T45299 CD0VI1 10412365 Ki > 100000 nM T45299 CJTH60 10432907 Ki = 844 nM T45299 C48HDV 10435701 Ki = 7700 nM T45299 CWG91R 10472893 Ki = 1700 nM T45299 CFS2U9 10474680 Ki = 35 nM T45299 C63GRO 10479438 IC50 = 70 nM T45299 CCP2N8 10480374 Ki > 8700 nM T45299 CV0X6G 10480463 IC50 > 11000 nM T45299 C7X1GS 10482360 IC50 = 390 nM T45299 CEI65Z 10483775 Ki = 1700 nM T45299 CS9NE0 10505479 IC50 > 30000000 nM T45299 CZA2C3 10521037 IC50 = 24000 nM T45299 C5ED3G 10529121 Ki = 36000 nM T45299 CU8N3V 10578280 Ki > 1000000 nM T45299 C2T4KP 10598728 IC50 = 250000 nM T45299 CI6WS3 10624333 IC50 = 5290 nM T45299 CEJ14F 10624997 Ki = 110000 nM T45299 C47FSO 10648183 IC50 = 9400 nM T45299 CPWH69 10648370 Ki > 1000000 nM T45299 CJG9H6 10669349 Ki = 19000 nM T45299 CW1G9B 10672666 IC50 > 10000 nM T45299 CP4QC5 10696511 Ki = 268000 nM T45299 CGYR23 10696955 Ki = 410000 nM T45299 CSK62G 10717029 IC50 = 34000 nM T45299 CIKF89 10719580 Ki = 84000 nM T45299 CZ0Q8K 10742217 Ki = 11000 nM T45299 C7RWD8 10744643 Ki = 29000 nM T45299 CLP31Y 10765317 IC50 = 1900 nM T45299 CKU82G 10791027 IC50 = 130000 nM T45299 CXLS49 10791461 IC50 = 62000 nM T45299 CWVK42 10814863 IC50 = 120000 nM T45299 C3IN8W 10815545 Ki = 180000 nM T45299 CVQE76 10816339 Ki = 190000 nM T45299 CLB15C 10871563 Ki = 210 nM T45299 CW7Q2U 10895700 IC50 > 2500 nM T45299 CQTC02 10903566 Ki = 2800 nM T45299 C8OA1L 10946869 Ki = 138000 nM T45299 C2TBO9 10959252 Ki = 3900 nM T45299 C43SNO 11004109 Ki = 690 nM T45299 CC39SB 11009950 Ki = 381000 nM T45299 CYZL25 11015002 Ki = 94 nM T45299 CD9WJ8 11057540 Ki = 160 nM T45299 C2Y6VW 11057779 Ki = 19 nM T45299 C3HNB2 11068806 Ki = 1300 nM T45299 CAD15G 11149953 Ki > 100000 nM T45299 C6LVG4 11186243 Ki = 8350 nM T45299 CTX9F3 11188793 Ki > 50000 nM T45299 CLA93S 11237163 Ki = 5502 nM T45299 CHLK70 11244460 Ki > 100000 nM T45299 CX9Z7A 11277660 IC50 > 250000 nM T45299 C86DZB 11292119 Ki = 1120 nM T45299 C91GMZ 11317532 Ki > 100000 nM T45299 C6CDN3 11347670 Ki = 83900 nM T45299 CLY5G8 11350400 Ki = 3130 nM T45299 CR8NW9 11351302 Ki > 20000 nM T45299 CTJ1Z2 11361949 Ki = 3950 nM T45299 CGW75B 11419694 Ki > 100000 nM T45299 CIQH43 11445130 IC50 = 250000 nM T45299 C9O4NF 11450922 IC50 > 62000 nM T45299 C63LIR 11473486 Ki = 2370 nM T45299 CJP9O1 11684611 Ki > 22000 nM T45299 CQ5U8H 11739438 Ki = 2320 nM T45299 C8GJO7 11754872 IC50 = 3990 nM T45299 CNPW05 11755188 IC50 > 10000 nM T45299 C7JLR1 11774107 Ki = 790 nM T45299 CR2E9T 11782463 Ki = 380 nM T45299 C98ZOR 11824040 Ki = 19000 nM T45299 CYX74A 11824584 Ki = 3000 nM T45299 C7VH6K 15950345 Ki > 35000 nM T45299 CA8Y1K 16046152 Ki = 23000 nM T45299 CNBJ60 16046153 Ki > 33000 nM T45299 C5TBL6 16049247 IC50 = 23000 nM T45299 C9BH4X 16086308 IC50 = 3100 nM T45299 CF1V2N 16086310 IC50 = 15000 nM T45299 C9JX7U 16086312 IC50 = 3400 nM T45299 CK7IM0 16086316 IC50 = 6600 nM T45299 CT9QM5 16086318 IC50 = 18000 nM T45299 CXO65R 16086320 IC50 = 3600 nM T45299 C3EUJ6 16086336 IC50 = 280 nM T45299 CR9EN3 16086338 IC50 = 4400 nM T45299 CR7B3D 16086340 IC50 = 13000 nM T45299 C90CXM 16086342 IC50 = 4300 nM T45299 C7T5AI 16086344 IC50 = 3700 nM T45299 CJZ63N 16086346 IC50 = 16000 nM T45299 C05XAN 16086348 IC50 = 5500 nM T45299 CACN42 16086349 IC50 = 6400 nM T45299 CN6CJ2 16220264 IC50 = 68510 nM T45299 CZB89F 16657876 Ki = 38000 nM T45299 CS9W6K 16657879 Ki > 100000 nM T45299 C09DTL 16657882 Ki > 100000 nM T45299 C3WX9G 16657950 Ki > 100000 nM T45299 CBPA54 16658031 Ki > 100000 nM T45299 C6V7DS 16658181 Ki > 100000 nM T45299 C0TW3X 16658183 Ki > 100000 nM T45299 CPNJ21 16658250 Ki = 23000 nM T45299 CG98OH 16658290 Ki = 108000 nM T45299 CO3ZV4 16658354 Ki > 30000 nM T45299 C46CDF 16658356 Ki > 100000 nM T45299 C8DI4G 16658357 Ki > 100000 nM T45299 C0Y4ZW 16658407 Ki > 100000 nM T45299 C6NR2O 16658408 Ki > 100000 nM T45299 CBX83S 16658633 Ki > 30000 nM T45299 CZ58FK 16658680 Ki > 30000 nM T45299 C70XKG 16658742 Ki > 100000 nM T45299 CQDT69 16658745 Ki > 100000 nM T45299 CU60AH 16718671 IC50 = 36600 nM T45299 COAB94 16718712 IC50 = 57000 nM T45299 CU28CE 16718713 IC50 = 6100 nM T45299 CLI4D7 16718757 IC50 = 3700 nM T45299 C2SFC0 16718759 IC50 = 4000 nM T45299 CC20PS 16718760 IC50 = 8000 nM T45299 CCKO80 16718762 IC50 = 44000 nM T45299 CTZ74D 16718807 IC50 = 125000 nM T45299 C37MRI 16718808 IC50 = 12000 nM T45299 CF4W5D 18727604 IC50 > 10000 nM T45299 CB0IQ4 18727607 IC50 > 11000 nM T45299 C31ZAL 18727831 IC50 > 11000 nM T45299 CJY67O 18727833 IC50 > 11000 nM T45299 C02HEA 18727834 IC50 > 11000 nM T45299 CJSL38 18727836 IC50 > 11000 nM T45299 C8AMY9 18727838 IC50 > 11000 nM T45299 CY8AC3 18727841 IC50 > 11000 nM T45299 CD02TK 18727852 IC50 > 11000 nM T45299 C1JMX5 18727855 IC50 > 11000 nM T45299 C24CAY 18771297 Ki = 126200 nM T45299 C2ID8R 20595260 IC50 > 10000 nM T45299 CMT46A 20595328 IC50 > 10000 nM T45299 C7LHE8 20641745 IC50 = 1850 nM T45299 CZ6KH9 20760195 Ki > 33000 nM T45299 CIM9C3 20801121 Ki > 100000 nM T45299 CC1Y0R 20801139 Ki > 100000 nM T45299 CS3HB4 20801160 Ki > 100000 nM T45299 C5UB8M 21705171 Ki = 367000 nM T45299 CA63IO 21706943 Ki = 7400 nM T45299 C80JYP 21707001 Ki = 18000 nM T45299 C3H6XW 21707065 Ki = 69110 nM T45299 C5JD2U 21707080 Ki = 27000 nM T45299 CI0SJ2 21967345 Ki > 8700 nM T45299 CN6P9I 22394409 Ki = 64010 nM T45299 CA3N9L 22883564 Ki > 8700 nM T45299 C1R0UD 22883585 Ki = 8700 nM T45299 C13-JAN 22883594 Ki > 8700 nM T45299 CQ70HF 23586156 IC50 = 173 nM T45299 CRX19I 23646295 Ki > 33000 nM T45299 CCRD27 23646312 Ki > 40000 nM T45299 C1WE6B 23646315 Ki > 33000 nM T45299 CSFH79 23646622 Ki = 360 nM T45299 C35HJA 23646623 Ki = 1700 nM T45299 C1L9VZ 23647194 Ki > 100000 nM T45299 CC29KT 23647198 Ki > 100000 nM T45299 CKH4O5 24180463 Ki > 21000 nM T45299 C7AYO1 24748789 IC50 = 16000 nM T45299 CVO5L6 24748791 IC50 = 68000 nM T45299 CUAY58 24749175 IC50 = 7000 nM T45299 CL2PU5 24750417 IC50 = 7300 nM T45299 CN0ZW3 24999867 Ki > 1000 nM T45299 CEM32W 25001205 Ki > 1000 nM T45299 C2H4PJ 25166809 Ki > 46000 nM T45299 CKM7Y8 25269170 Ki > 20000 nM T45299 C9OMR4 44264598 Ki > 200000 nM T45299 C9RND0 44264660 Ki > 200000 nM T45299 CL7NY5 44274017 IC50 > 10000 nM T45299 CMG90C 44274089 IC50 > 10000 nM T45299 C19OGX 44278104 Ki = 632 nM T45299 CQ82ZW 44286426 IC50 > 2500 nM T45299 COPR02 44286428 IC50 > 2500 nM T45299 CS5U7F 44286453 IC50 > 2500 nM T45299 C8APX2 44290947 Ki > 8700 nM T45299 CJU7B0 44298507 Ki = 60100 nM T45299 CS1I3Q 44298510 Ki = 258500 nM T45299 C2P7QZ 44298511 Ki = 342000 nM T45299 COU03N 44298523 Ki = 71500 nM T45299 C13TMY 44298524 Ki = 53800 nM T45299 CRS39A 44298525 Ki = 65900 nM T45299 C29MVU 44303719 Ki > 95000 nM T45299 C3FB4I 44303721 Ki > 95000 nM T45299 CQLA16 44303733 Ki > 95000 nM T45299 C5RZL0 44303743 Ki = 880 nM T45299 CTE75P 44303769 Ki = 2000 nM T45299 C16GOI 44303778 Ki = 2400 nM T45299 C26ZUK 44303789 Ki = 9400 nM T45299 CN6V9A 44303803 Ki = 3600 nM T45299 C67ZRW 44303804 Ki = 53000 nM T45299 CB38WA 44303805 Ki = 1800 nM T45299 CL0U1A 44303806 Ki = 3900 nM T45299 CVO2D9 44303808 Ki = 94000 nM T45299 C0JZY5 44303810 Ki = 21000 nM T45299 CFJ4W3 44303811 Ki = 6900 nM T45299 CE0R9A 44303824 Ki > 95000 nM T45299 C5YF7O 44303839 Ki > 95000 nM T45299 C2LY4T 44303843 Ki = 1500 nM T45299 C3HXW6 44303858 Ki = 35 nM T45299 CYW9S8 44303912 Ki > 563000 nM T45299 CIQZ37 44303925 Ki = 300000 nM T45299 CJN72A 44303933 Ki = 1700 nM T45299 CXCY31 44303935 Ki = 150000 nM T45299 C4SN8T 44304006 Ki > 95000 nM T45299 CL16JC 44304046 Ki > 95000 nM T45299 CAM6R0 44304047 Ki > 95000 nM T45299 CR4V0L 44304084 Ki = 225000 nM T45299 CG37DH 44304086 Ki = 506000 nM T45299 C7UJH1 44304087 Ki = 338000 nM T45299 CG0R8N 44304097 Ki = 181000 nM T45299 CJ80KE 44304098 Ki > 95000 nM T45299 CG8TI6 44304099 Ki > 95000 nM T45299 C9W8QC 44304100 Ki > 563000 nM T45299 CE31BF 44304104 Ki > 95000 nM T45299 C9XIO1 44304105 Ki > 95000 nM T45299 C83YIU 44304139 Ki = 258000 nM T45299 CP5S9K 44304192 Ki = 95000 nM T45299 CKD98A 44304353 Ki > 95000 nM T45299 CZEX59 44311229 IC50 > 33000 nM T45299 CKP5W7 44311564 IC50 > 1100 nM T45299 CAG6M5 44327046 Ki = 5600 nM T45299 C26KJP 44330423 Ki = 1100 nM T45299 CW1XE9 44330628 Ki = 280 nM T45299 C1Z5FA 44330631 Ki = 51 nM T45299 CK8FJ6 44330632 Ki = 7000 nM T45299 CS1V3W 44330665 Ki = 3800 nM T45299 CWV7X5 44330835 Ki = 750 nM T45299 C98KLH 44330847 Ki = 3370 nM T45299 CSM3B6 44330879 IC50 > 180000 nM T45299 CE69GW 44331194 IC50 = 180000 nM T45299 C7Y8IG 44334488 Ki = 1600 nM T45299 CHL01I 44334805 Ki = 130 nM T45299 C8BKP0 44335014 IC50 = 430000 nM T45299 CRT4G3 44335601 Ki = 20000 nM T45299 C7Z9WL 44335624 Ki = 470000 nM T45299 CQ37SV 44339192 Ki = 123900 nM T45299 CCA37E 44339231 Ki = 128500 nM T45299 C89EZV 44339232 Ki = 159200 nM T45299 C8JQA9 44339233 Ki = 140100 nM T45299 C3XI4S 44339270 Ki = 123900 nM T45299 C98MCJ 44339277 Ki = 95100 nM T45299 C7RVG9 44343560 IC50 = 2100 nM T45299 CXRS15 44343561 IC50 = 2500 nM T45299 CR7BU3 44343575 IC50 = 2300 nM T45299 CUTB94 44343630 IC50 = 6100 nM T45299 CL5IB0 44343631 IC50 = 5800 nM T45299 COE8Y7 44343829 IC50 = 14900 nM T45299 C17JVH 44343830 IC50 = 3800 nM T45299 CR1O2L 44343833 IC50 = 3220 nM T45299 C8SR3D 44343849 IC50 = 9000 nM T45299 CKS43F 44343885 IC50 = 2200 nM T45299 CLCX01 44343886 IC50 = 7200 nM T45299 CAY34C 44347478 Ki = 436000 nM T45299 CT0QN1 44347480 Ki = 746000 nM T45299 C1UN9I 44347534 Ki > 1000000 nM T45299 C0V2FL 44347624 Ki > 500000 nM T45299 CX9MJ6 44356715 Ki = 120 nM T45299 C81XMY 44358802 IC50 = 48000 nM T45299 CPX09V 44358866 IC50 > 30000000 nM T45299 CSNJ26 44358867 IC50 > 30000000 nM T45299 CL0U6H 44358868 IC50 > 30000000 nM T45299 CUE9P4 44359039 IC50 = 23000 nM T45299 C2NQC0 44359053 IC50 = 900 nM T45299 C7IJY6 44367340 Ki = 950 nM T45299 C5SD9G 44367355 Ki = 69000 nM T45299 C8YP2H 44367372 Ki = 980 nM T45299 CWD01E 44367382 Ki = 70000 nM T45299 CXB28Z 44367430 Ki = 23000 nM T45299 CFY5B6 44367435 Ki = 33000 nM T45299 CYDQ04 44367444 Ki = 120000 nM T45299 C34XTM 44375987 IC50 = 329 nM T45299 CD0W7C 44376100 IC50 = 1880 nM T45299 C0Y8QD 44376252 IC50 = 740 nM T45299 C5R2PM 44376328 IC50 = 9960 nM T45299 C5VDG0 44376417 IC50 = 150 nM T45299 CG64YQ 44376426 IC50 = 4010 nM T45299 CD36KV 44380417 Ki = 6700000 nM T45299 C9SD3E 44383242 Ki > 8700 nM T45299 C43KTU 44383519 Ki > 8700 nM T45299 CG7LT1 44385488 IC50 > 11000 nM T45299 C94GZU 44385541 IC50 > 11000 nM T45299 C3T9XK 44385607 IC50 > 11000 nM T45299 CKY0P4 44385611 IC50 > 11000 nM T45299 CUS20V 44385673 IC50 > 11000 nM T45299 CZ8XL6 44385679 IC50 > 11000 nM T45299 COQH07 44385725 IC50 > 2500 nM T45299 CL5BA4 44385729 IC50 > 11000 nM T45299 C3DSN7 44385768 IC50 > 11000 nM T45299 C8USN9 44385769 IC50 > 11000 nM T45299 CX9W5Z 44385770 IC50 > 2500 nM T45299 C2E8DS 44385771 IC50 > 11000 nM T45299 C2VFC6 44385772 IC50 > 11000 nM T45299 CN8V0W 44385779 IC50 > 11000 nM T45299 C7MXA5 44385833 IC50 > 2500 nM T45299 CBEA65 44385842 IC50 > 11000 nM T45299 CC9M7E 44385869 IC50 > 11000 nM T45299 C8WK4A 44385891 IC50 > 11000 nM T45299 C3D2CL 44385935 IC50 > 11000 nM T45299 CW08OY 44385998 IC50 > 11000 nM T45299 C8F2RG 44386052 IC50 > 2500 nM T45299 CV6KG4 44386059 IC50 > 11000 nM T45299 CGU69V 44386179 IC50 > 11000 nM T45299 CS65LH 44386185 IC50 > 11000 nM T45299 C5YF1O 44386205 IC50 > 2500 nM T45299 CU0P5T 44386242 IC50 > 11000 nM T45299 CU9J0D 44386250 IC50 > 11000 nM T45299 C9G7QW 44386322 IC50 > 11000 nM T45299 C31CUG 44386326 IC50 > 11000 nM T45299 C52MCK 44386366 IC50 > 2500 nM T45299 C2WCE4 44386371 IC50 > 11000 nM T45299 C52POK 44386417 IC50 > 11000 nM T45299 CRX1I9 44386418 IC50 > 11000 nM T45299 CBG1U6 44386478 IC50 > 2500 nM T45299 CIBD76 44386484 IC50 > 11000 nM T45299 C8ME4O 44386493 IC50 > 11000 nM T45299 CD4AH3 44386540 IC50 > 11000 nM T45299 CHAO48 44386542 IC50 > 11000 nM T45299 CLNO15 44386637 IC50 > 11000 nM T45299 C81IMH 44386642 IC50 > 11000 nM T45299 CWTU45 44386804 IC50 > 2500 nM T45299 C4JB0M 44386841 IC50 > 11000 nM T45299 CA0W2K 44386893 IC50 > 2500 nM T45299 C5MR1F 44386934 IC50 > 11000 nM T45299 CA45DZ 44387044 IC50 > 11000 nM T45299 C39LUW 44387104 IC50 > 11000 nM T45299 C2QD1K 44387206 IC50 > 11000 nM T45299 CAY27D 44392382 Ki = 10430 nM T45299 C2SQ1C 44392401 Ki = 5590 nM T45299 C4VKE9 44392403 Ki > 50000 nM T45299 CYL52J 44392413 Ki = 5049 nM T45299 CN8CJ3 44392416 Ki = 30783 nM T45299 CE42KB 44392423 Ki = 5786 nM T45299 CORK28 44392427 Ki = 21924 nM T45299 CP67EA 44411094 IC50 = 125 nM T45299 CM8OZ0 44411137 IC50 = 687 nM T45299 CPN1S0 44416248 IC50 = 8600 nM T45299 CVO5Q1 44432538 Ki > 20000 nM T45299 C2SMQ6 44433791 Ki > 1000000 nM T45299 CR16BF 44434808 Ki > 21000 nM T45299 CQIX73 44434809 Ki > 21000 nM T45299 C5R8HJ 44434815 Ki > 21000 nM T45299 COG34X 44434818 Ki > 21000 nM T45299 C9T1DP 44434835 Ki > 21000 nM T45299 C30CFX 44436704 IC50 = 44000 nM T45299 CB86HU 44453827 IC50 = 29 nM T45299 C8Z4WO 44459967 IC50 = 851.14 nM T45299 C86ORE 44459987 IC50 = 1288.25 nM T45299 CVZW52 44537923 IC50 = 3100 nM T45299 C8XT1U 44626341 IC50 = 5200 nM T45299 C7JP5Q 44626343 IC50 > 30000 nM T45299 CDG17C 44626344 IC50 = 14000 nM T45299 C6I0TN 44626345 IC50 = 8500 nM T45299 CGXD19 45485586 IC50 = 3900 nM T45299 C9OZ8H 45485587 IC50 = 18000 nM T45299 C0H5ST 45485592 IC50 > 30000 nM T45299 CPT2Y1 45485611 IC50 = 15000 nM T45299 C27HKO 45485622 IC50 = 22000 nM T45299 C3HKP7 45485641 IC50 = 16000 nM T45299 CHT06J 45485667 IC50 > 30000 nM T45299 C76CDZ 45485668 IC50 = 10000 nM T45299 CGX93B 45485669 IC50 = 11000 nM T45299 C0R4EB 45485670 IC50 = 28000 nM T45299 CI5EJ4 45485671 IC50 > 30000 nM T45299 CCG5U1 46196561 Ki > 60000 nM T45299 CA6GQ5 53341037 Ki > 6150 nM T45299 CIKQ81 53345652 Ki > 130 nM T45299 CXWS90 53345968 Ki > 1000 nM T45299 CV60BK 53488415 Ki = 1279 nM T45299 C8U4OD 56649692 IC50 > 1000000 nM T45299 CLU95A 57325502 IC50 = 26000 nM T45299 CV42AN 57390824 IC50 = 21000 nM T45299 C1GIV7 57390825 IC50 = 8600 nM T45299 CM7FT5 57390879 IC50 = 11000 nM T45299 CXV4U9 57394359 IC50 = 3400 nM T45299 CIC2U6 57397927 IC50 = 5700 nM T45299 C98KRU 57397928 IC50 = 9700 nM T45299 CBKD41 57400356 IC50 = 13000 nM T45299 CKV6R8 57401327 IC50 = 5300 nM T45299 CES6D2 57403083 IC50 = 8400 nM T45299 C3RZ8G 57404502 IC50 = 200000 nM T45299 CVWP51 57404503 IC50 > 190000 nM T45299 C9XW1C 57842830 Ki > 10000 nM T45299 C60HCV 57976401 Ki > 6150 nM T45299 CHB27Y 57976410 Ki = 10500 nM T45299 CM8UJ7 57976444 Ki = 19000 nM T45299 CQ71KE 57976446 Ki = 17000 nM T45299 CSC0L5 59020200 Ki > 43000 nM T45299 C91APY 59095797 IC50 > 33000 nM T45299 C69SED 59095888 IC50 > 33000 nM T45299 CPW2H7 59315536 Ki > 10000 nM T45299 CO38AC 59402011 Ki > 46000 nM T45299 CE5A7B 60162406 Ki > 100000 nM T45299 CWOD93 66744646 Ki > 6150 nM T45299 CKWQ82 67155200 Ki = 3600 nM T45299 CPO6Z9 69496614 IC50 = 1850 nM T45299 C1DUV4 69496716 IC50 > 30000 nM T45299 C6YW5E 69496717 IC50 = 470 nM T45299 CUG9Z7 69496724 IC50 = 1450 nM T45299 CR59OP 69496744 IC50 = 1600 nM T45299 CX97VL 69496820 IC50 = 1580 nM T45299 CD5ZW0 69496838 IC50 = 5700 nM T45299 C6AU1R 70252985 Ki > 14700 nM T45299 CTO5I6 70253788 Ki > 14700 nM T45299 CL4RK8 70683232 IC50 > 250000 nM T45299 CX0VK6 70689516 IC50 > 250000 nM T45299 C2UOG4 70693724 IC50 > 250000 nM T45299 CE27BR 70695842 IC50 > 250000 nM T45299 C9EL3C 71260387 Ki > 6150 nM T45299 C45SHM 71451304 Ki > 20000 nM T45299 CJPF90 71548883 Ki > 6200 nM T45299 C30ZKJ 71561420 Ki > 40000 nM T45299 C62ZTJ 71660643 IC50 > 33000 nM T45299 C78DJQ 71711730 IC50 < 10000 nM T45299 CD53RA 71716975 Ki > 120000 nM T45299 CSP5T2 71716976 Ki > 120000 nM T45299 CM83VP 72163524 IC50 > 10000 nM T45299 CRBH34 72164200 IC50 > 33000 nM T45299 CWNZ45 72164201 IC50 > 33000 nM T45299 CLI36U 72551247 Ki = 9100 nM T45299 CB8RP9 73350124 IC50 = 30000 nM T45299 CL8EG7 73350757 Ki = 113 nM T45299 CMD5V7 86583041 Ki > 21900 nM T45299 CWP85J 87360663 IC50 = 32000 nM T45299 CO6U9I 88582319 Ki = 10100 nM T45299 C65TLW 101862198 Ki > 1000000 nM T45299 CHQ5P7 118987013 Ki > 21900 nM T45299 CK0W2P 127027635 Ki > 8600 nM T45299 CJ6DA9 127028140 IC50 > 10000 nM T45299 CD9KI3 127028141 IC50 > 10000 nM T45299 CPC0M8 127031390 Ki > 21900 nM T45299 C1BWV2 127035672 Ki > 1000000 nM T45299 CVRY56 127036086 Ki > 1000000 nM T45299 C9B6LT 127037264 Ki > 1000000 nM T45299 C60HLK 127037469 Ki > 1000000 nM T45299 C85ROH 127041472 IC50 > 100000 nM T45299 CT2RV6 134130781 IC50 > 1000000 nM T45299 CWV3G6 134131077 IC50 > 200000 nM T45299 CS8FV1 134131084 IC50 > 200000 nM T45299 C92RTL 134131303 IC50 > 200000 nM T45299 CL37SG 134131589 IC50 > 200000 nM T45299 C6HTD5 135393470 IC50 > 10000 nM T45299 C7NA6E 135393474 IC50 > 20000 nM T45299 CD53CZ 135404951 Ki = 7700 nM T45299 C5XA6H 135407717 Ki = 48000 nM T45299 C0OX6T 135407736 Ki = 56000 nM T45299 C61XOA 135427245 Ki = 69000 nM T45299 C8WS4O 135443730 Ki = 113000 nM T45299 CTP5V8 135444609 Ki = 1000 nM T45299 C4M5BF 135450980 Ki = 19000 nM T45299 CDT1C6 135452907 Ki = 360 nM T45299 C3YT2M 135452929 Ki = 3900 nM T45299 CPN5I3 135452944 Ki = 3 nM T45299 C9KLD3 135455964 Ki > 8700 nM T45299 CJWC64 135462427 Ki = 1070 nM T45299 C5O6JX 135469686 Ki = 6 nM T45299 C9XMA6 135469687 Ki = 150 nM T45299 CXS6B9 135471524 Ki = 25000 nM T45299 C2PFI8 135475618 Ki = 14000 nM T45299 CG2N5B 135484079 Ki = 20 nM T45299 CBE9G0 135490854 Ki = 31000 nM T45299 CPW07U 135493126 Ki = 480 nM T45299 CMQ6O0 135501618 Ki = 69000 nM T45299 CVA61N 135512760 Ki = 41000 nM T45299 CLFR21 135528485 Ki = 165000 nM T45299 CHEQ21 135528490 Ki = 3200 nM T45299 CK97FT 135533257 Ki = 280 nM T45299 CAD75F 135535997 Ki = 150000 nM T45299 CCH49A 135544551 Ki = 10000 nM T45299 CKLD47 135544579 Ki = 100000 nM T45299 C8KNC4 135681488 Ki = 6 nM T45299 C91UXW 135802775 Ki > 8700 nM T45299 C6S5OL 136034781 Ki = 225000 nM T45299 CYQ70K 136053621 IC50 > 11000 nM T45299 CN70IU 136092208 Ki > 75000 nM T45299 C5N3KP 136092209 Ki = 71000 nM T45299 C1BUH6 136092210 Ki = 263000 nM T45299 CFQ2C8 136092211 Ki = 150000 nM T45299 CX5R9J 136092212 Ki = 425000 nM T45299 C35PXN 136092213 Ki = 33000 nM T45299 CEXJ30 136092214 Ki > 75000 nM T45299 CS6QH0 136092215 Ki = 29000 nM T45299 CMR7L4 136092216 Ki = 275000 nM T45299 CN0WR7 136092217 Ki = 45000 nM T45299 COCN35 136092218 Ki = 44000 nM T45299 CA79JC 136092219 Ki = 3200 nM T45299 CPK6X2 136198635 Ki = 2700 nM T45299 CRJ5S4 136198636 Ki = 7500 nM T45299 C7WE2G 136198637 Ki = 8700 nM T45299 C12UWY 136198638 Ki = 8700 nM T45299 C26ZPI 136264091 IC50 > 250000 nM T45299 C8VJW4 136266885 IC50 = 200000 nM T45299 CC0BI4 136268735 IC50 > 250000 nM T45299 CO51HN 139030452 IC50 > 20000 nM T45299 CX07YE 139592452 Ki > 6150 nM T45299 CE6C0A 145970642 Ki = 994 nM T45299 C4HLX8 146029523 IC50 > 20000 nM T45299 CICU31 155511394 Ki = 2834 nM T45299 C2VX3G 155512946 Ki = 2940 nM T45299 C2CI8S 155513907 Ki = 3525 nM T45299 CYT20V 155514020 Ki > 50000 nM T45299 CAT98N 155514640 Ki > 10000 nM T45299 CF96DM 155518671 Ki > 10000 nM T45299 C7DUX3 155520916 Ki > 10000 nM T45299 C46AZL 155530642 Ki > 25000 nM T45299 CL90DN 155540666 Ki > 10000 nM T45299 C4P2GV 155543617 Ki > 25000 nM T45299 CU9FL4 155551858 Ki > 50000 nM T45299 CU8LR3 155555208 Ki > 25000 nM T45299 CP4F1U 155567613 Ki > 50000 nM T45299 CEZ8B9 155568406 Ki > 50000 nM T45299 CVK8X3 44338049 IC50 = 0.7 nM T45299 CD81GH 46830813 IC50 > 2500 nM T45299 D00KJP 10322586 Ki = 8600 nM T45299 D00PEJ 16658631 Ki = 15000 nM T45299 D00POF 21707121 Ki = 34564 nM T45299 D01JUI 44339119 Ki = 19000 nM T45299 D01LCS 447480 Ki = 690 nM T45299 D02AVL 18376720 Ki > 5000 nM T45299 D02PAU 16731825 Ki > 5000 nM T45299 D02YIW 1794 IC50 > 10000 nM T45299 D03ZUM 6917805 IC50 = 950 nM T45299 D06AVE 10200844 Ki = 6230 nM T45299 D06CJP 16658353 Ki > 100000 nM T45299 D06HOI 44249821 Ki = 3700 nM T45299 D06MTX 1506 Ki = 75000 nM T45299 D07SFI 2332 Ki = 910000 nM T45299 D09YLF 44339283 Ki = 13000 nM T45299 D09YQM 9802488 IC50 > 8250 nM T45299 D0A8WP 447732 Ki = 31800 nM T45299 D0C3QE 21192457 Ki = 13000 nM T45299 D0F6EZ 44436702 Ki > 1000000 nM T45299 D0J1CC 11948634 Ki > 10000 nM T45299 D0J1QT 44473100 Ki = 665 nM T45299 D0JU9N 6914623 Ki > 2800 nM T45299 D0K0GU 44392430 Ki = 4465 nM T45299 D0K4PK 16658352 Ki = 24000 nM T45299 D0K7YL 447476 Ki = 35 nM T45299 D0MQ6K 10574241 Ki > 10000 nM T45299 D0ON2Z 204102 Ki > 2300 nM T45299 D0R9CH 3400921 Ki > 5000 nM T45299 D0S4MQ 44392405 Ki = 13380 nM T45299 D0Y8QU 9869156 IC50 > 2500 nM T50429 D03HJK 447043 IC50 > 10000000 nM T50429 D07QCE 2265 IC50 = 8100000 nM T50429 D08LTU 54675783 Ki = 180000 nM T50429 D08ROP 3899 IC50 = 2400000 nM T50429 D0AO5H 5578 IC50 = 7500000 nM T50429 D0C4YC 4075 IC50 > 10000000 nM T50429 D0D4CY 5336 IC50 > 10000000 nM T50429 D0N0EQ 19649 Ki = 560000 nM T50429 D0R0ZL 446598 IC50 = 5100000 nM T50429 D0R6RC 54675777 IC50 = 100000 nM T50429 D0R9OH 5329 IC50 > 10000000 nM T50429 D0S0LZ 54671203 Ki = 630000 nM T50429 D0SV8E 126941 IC50 > 10000000 nM T50429 CFB4W1 253688 IC50 = 1000 nM T50429 C1HYD5 265935 IC50 = 3300 nM T50429 CA17WJ 3562756 IC50 > 10000000 nM T50429 CZ60QE 6501454 Ki = 183000 nM T50429 C7KQ3Z 11589584 IC50 = 21000 nM T50429 C0U7YP 13891339 IC50 = 240 nM T50429 C3PQ2R 35429407 Ki = 1430000 nM T50429 CUR3G8 47013852 Ki = 4643000 nM T50429 CE75GT 47164586 Ki = 632000 nM T50429 CTE72N 51049631 IC50 = 560 nM T50429 CLTR59 54756931 IC50 = 500000 nM T50429 C58RGE 54756933 IC50 = 230000 nM T50429 C09ESA 54756935 IC50 = 19000 nM T50429 C46XLD 54756937 IC50 = 12000 nM T50429 C1MFN2 54756939 IC50 = 400 nM T50429 COF2G6 54756941 IC50 = 2400 nM T50429 CLZX23 54758326 IC50 > 1000000 nM T50429 CFR5O6 54758328 IC50 > 1000000 nM T50429 CV6C2Q 54758330 IC50 > 500000 nM T50429 C3RIP0 54758419 IC50 = 310000 nM T50429 C1MQ7C 54758421 IC50 = 2100000 nM T50429 CRB3E9 54758423 IC50 = 310000 nM T50429 CHU30Y 54758425 IC50 > 1000000 nM T50429 CGI1E2 54758427 IC50 > 1000000 nM T50429 C4KZC9 54758429 IC50 > 1000000 nM T50429 CC62WY 86340175 IC50 = 50 nM T50429 C72DTE 122702847 IC50 = 79.43 nM T50429 CF89UM 122702852 IC50 = 100 nM T50429 C2K6ZF 122702937 IC50 = 50.12 nM T50429 CO98AS 122702951 IC50 = 39.81 nM T50429 C5QKE4 122702999 IC50 = 158.49 nM T50429 CA7QO4 122703166 IC50 = 125.89 nM T50429 C8WD7Q 126601763 Ki = 488000 nM T50429 CG09SE 126601779 Ki = 2823000 nM T50429 C7D9YU 126601789 Ki > 10000000 nM T50429 C0T8LJ 126601811 Ki > 10000000 nM T50429 C9X5PA 126601948 Ki > 10000000 nM T50429 C6SU3Z 126615756 Ki = 180000 nM T50429 CI3C4Q 126616118 Ki = 591000 nM T50429 CRGE48 134308661 Ki = 47000 nM T50429 C3UG2Q 137644769 Ki = 64000 nM T50429 C05MLZ 137661236 Ki = 88000 nM T50429 CA3MW0 145981940 IC50 = 29000 nM T50429 CPJ12Q 145987120 IC50 = 16000 nM T50429 C2TM5J 145989141 IC50 = 21000 nM T50429 C2JXT5 145993007 IC50 = 190000 nM T50429 C7G9WS 145993776 IC50 = 36000 nM T50429 CH69FL 146680924 IC50 = 28000 nM T50429 C54VSY 155515570 IC50 = 36000 nM T50429 C1VN8A 155520618 IC50 = 8800 nM T50429 C7CU2H 155528540 IC50 = 129000 nM T50429 CH5VR7 155530421 IC50 = 39000 nM T50429 C6VO9W 155536240 IC50 = 53000 nM T50429 CDY59I 155553395 IC50 = 22000 nM T50429 CZR6D8 155553413 IC50 = 64000 nM T50429 D01FNC 21771691 IC50 = 640 nM T50429 D02ZNQ 5298 IC50 = 2500 nM T50429 D0YP0A 24970878 IC50 = 3400 nM T48040 CUB4P8 1007407 IC50 = 11500 nM T48040 C2CDW6 5346781 IC50 > 50000 nM T48040 CZJR62 5346811 IC50 = 12000 nM T48040 C28ITK 5760065 IC50 = 9600 nM T48040 CDG1C7 5931617 IC50 = 17800 nM T48040 CRGW50 5990731 IC50 = 6800 nM T48040 C7Q3ZW 6104209 IC50 = 13100 nM T48040 C6MW9G 11836699 IC50 = 9100 nM T48040 C9KF7H 24893997 IC50 > 50000 nM T48040 C2NVS6 24893998 IC50 > 50000 nM T48040 CB1QI9 30135276 IC50 > 50000 nM T48040 CY3FQ9 45105371 IC50 = 4820 nM T48040 C9DWJ8 45105373 IC50 = 12600 nM T48040 C7P8AZ 50883606 IC50 = 1930 nM T48040 CC09QH 50884279 IC50 = 1600 nM T48040 C0W8LM 50884438 IC50 = 5230 nM T48040 CK6AQ0 50885828 IC50 = 820 nM T48040 C6MLP7 50885855 IC50 = 1300 nM T48040 C32GWL 132169606 IC50 = 14100 nM T48040 C0OLY5 132169617 IC50 = 9100 nM T48040 CZ68VJ 132169621 IC50 = 14300 nM T48040 CS56EJ 132169626 IC50 = 12000 nM T48040 CW6MT7 132169645 IC50 > 50000 nM T48040 CE8DW6 132169659 IC50 = 11700 nM T48040 CCZ76J 132169682 IC50 >= 25000 nM T48040 CJPU46 132169683 IC50 = 13400 nM T48040 C5XZ3P 132169738 IC50 = 11900 nM T48040 CAL1C0 132169746 IC50 > 50000 nM T48040 CB6EQ0 132169827 IC50 > 50000 nM T48040 CZP71S 132169832 IC50 >= 25000 nM T48040 CDB5R9 132169876 IC50 = 9100 nM T48040 CT6OS9 132169899 IC50 = 9800 nM T48040 CGIA39 132169908 IC50 = 8400 nM T48040 CB03OA 132178937 IC50 > 25000 nM T21585 D09JEJ 24748573 IC50 = 41 nM T21585 D0E3TC 44259 IC50 = 1310 nM T21585 D05BVP 3232621 IC50 = 6936 nM T21585 D09CDR 77105816 IC50 = 190 nM T21585 D0CC7E 77105818 IC50 = 320 nM T21585 D0JQ0Z 46916176 IC50 = 435 nM T21585 CU80LI 3233012 IC50 = 8744 nM T21585 CGAT36 5327151 IC50 > 1000 nM T21585 CACS26 11561968 Ki > 2000 nM T21585 CP04JC 11666231 IC50 = 86.6 nM T21585 CU0E8O 11690457 Ki > 2000 nM T21585 CR3BS0 12248905 IC50 = 1800 nM T21585 CGLQ20 44223952 IC50 = 7448 nM T21585 CR6VH2 44223953 IC50 = 6555 nM T21585 C2IBW0 44223954 IC50 > 10000 nM T21585 CS3Q2Y 44223955 IC50 = 3294 nM T21585 C5M1UN 44223957 IC50 > 10000 nM T21585 CK8G1T 44223965 IC50 = 2017 nM T21585 CJ8KD4 44223966 IC50 > 10000 nM T21585 CCW0V4 44223967 IC50 > 10000 nM T21585 CF78WD 44223968 IC50 > 10000 nM T21585 CNE30X 44223970 IC50 = 1924 nM T21585 CYR45S 44223971 IC50 = 4655 nM T21585 CLZ62P 44223973 IC50 = 4949 nM T21585 CIXB09 44223974 IC50 = 6450 nM T21585 C2OBX8 44223977 IC50 = 4650 nM T21585 C3JBN1 44968184 IC50 > 10000 nM T21585 CYW79D 44968186 IC50 = 6172 nM T21585 C5OYK3 44968199 IC50 > 10000 nM T21585 C2T0EM 44968221 IC50 > 10000 nM T21585 C8NA2J 44968224 IC50 > 10000 nM T21585 CR8DC5 44968225 IC50 > 10000 nM T21585 CV19YK 44968230 IC50 > 10000 nM T21585 CD4ZN1 44968231 IC50 > 10000 nM T21585 C15EJK 46916169 IC50 > 10000 nM T21585 CHG8C4 46916170 IC50 = 3527 nM T21585 CI56BA 46916172 IC50 = 3019 nM T21585 CZ5DJ4 46916177 IC50 = 2556 nM T21585 CXK37B 46916178 IC50 = 3642 nM T21585 CL1GW0 46916179 IC50 = 1320 nM T21585 CZ6DK4 46916182 IC50 = 5461 nM T21585 C9NC6W 46926516 IC50 > 10000 nM T21585 CZ1D2A 46926518 IC50 = 1473 nM T21585 C7S6HT 46926519 IC50 > 10000 nM T21585 CPE98Z 46926523 IC50 = 3634 nM T21585 C0IVD1 46926527 IC50 = 3232 nM T21585 C7T5HW 49795865 IC50 = 2663 nM T21585 C6N8EY 49795866 IC50 = 2934 nM T21585 C5EWG8 49855158 IC50 > 10000 nM T21585 CS6N8Z 54581884 IC50 > 10000 nM T21585 CW9AE7 60034150 IC50 > 1000 nM T21585 C1MR8Q 60097495 IC50 > 1000 nM T21585 CV63UL 67240318 IC50 > 10000 nM T21585 C21JAS 76853169 IC50 = 7000 nM T21585 CU04XY 77105624 IC50 > 10000 nM T21585 CTIA65 77105820 IC50 = 8000 nM T21585 CKB1P9 77106023 IC50 = 180 nM T21585 CXYW85 77106025 IC50 > 10000 nM T21585 C2UDS0 77106026 IC50 > 10000 nM T21585 C97SJD 77106027 IC50 = 6100 nM T21585 CFQ10R 77106028 IC50 = 710 nM T21585 CO14DP 77106030 IC50 = 7000 nM T21585 C9G3PA 77106234 IC50 = 6100 nM T21585 CPD27I 77106235 IC50 > 10000 nM T21585 CLOR37 77106236 IC50 > 10000 nM T21585 C2GLD8 77106237 IC50 = 6800 nM T21585 C0GYK1 86765296 IC50 = 2300 nM T21585 C3KJ8R 98073446 IC50 = 530 nM T21585 C2LWZ1 129318964 IC50 = 5590 nM T21585 C4Z5MQ 131839619 IC50 > 1000 nM T21585 C4QM9O 134397095 IC50 > 1000 nM T21585 CQ1K2W 134397387 IC50 > 1000 nM T21585 CR08AO 134397388 IC50 > 1000 nM T21585 CIN73J 134397390 IC50 > 1000 nM T21585 C6I1YX 134397391 IC50 > 1000 nM T21585 CQ9D1Z 134397392 IC50 > 1000 nM T21585 CUX8N5 134397449 IC50 > 1000 nM T21585 CDC39N 134397450 IC50 > 1000 nM T21585 C8RN6W 134397451 IC50 > 1000 nM T21585 CE1HY2 134397452 IC50 > 1000 nM T21585 CIR51J 134397453 IC50 > 1000 nM T21585 C72KFM 134397463 IC50 > 1000 nM T21585 CT16YX 134397502 IC50 > 1000 nM T21585 CI45HZ 134397798 IC50 > 1000 nM T21585 C5J2WV 138728749 IC50 > 10000 nM T21585 CVU63L 139582016 IC50 > 10000 nM T21585 C8PH9S 139582017 IC50 > 10000 nM T21585 CX05ZN 145979845 IC50 > 10000 nM T21585 C2MD1Q 155513187 IC50 > 10000 nM T21585 D06CXU 46926513 IC50 > 10000 nM T21585 D07OCA 5330812 IC50 = 29.2 nM T21585 D0D2FC 2794188 IC50 > 1000 nM T21585 D0UI7U 46926514 IC50 > 10000 nM T04831 D0E3TC 44259 IC50 < 100 nM T04831 CGAN35 2856 IC50 = 16000 nM T04831 C18WEB 490561 IC50 < 100 nM T04831 CYZU17 937050 IC50 = 13000 nM T04831 CLG63C 1530863 IC50 = 9400 nM T04831 CZ5KB1 2455709 IC50 = 12000 nM T04831 CVB83T 5330811 IC50 = 8000 nM T04831 C2NP5X 6897738 IC50 = 11000 nM T04831 C2WG8I 7216437 IC50 = 11000 nM T04831 C7L3JN 9124464 IC50 = 13000 nM T04831 C5B3XJ 11620410 IC50 > 40000 nM T04831 CV56YS 16414650 IC50 = 20000 nM T04831 CQOT74 16805560 IC50 = 15000 nM T04831 CJCQ86 17395684 IC50 = 19000 nM T04831 C6QT0J 44622837 IC50 > 1000 nM T04831 CU9GM5 53307873 Ki = 3400 nM T04831 CXB94H 53466728 IC50 > 10000 nM T04831 CYQ41S 53466951 IC50 = 978 nM T04831 CX0R1K 53469059 IC50 = 905 nM T04831 CV7C0D 53469060 IC50 = 359 nM T04831 CCKD45 53469061 IC50 = 99 nM T04831 C91STB 53469449 IC50 = 291 nM T04831 CZ1CI3 53469824 IC50 > 10000 nM T04831 CQEA01 56659460 IC50 > 100000 nM T04831 C5KEW0 56659461 IC50 = 3000 nM T04831 C7PCY5 56659462 IC50 > 100000 nM T04831 C1JD8Z 56659512 IC50 = 12000 nM T04831 C34VCR 56659514 IC50 = 90000 nM T04831 CPQ2A9 56659515 IC50 = 9000 nM T04831 CYK40N 56659516 IC50 > 100000 nM T04831 C39BXF 56659517 IC50 = 600 nM T04831 CD65YZ 56662919 IC50 = 1500 nM T04831 C6MR1L 56662961 IC50 = 1500 nM T04831 C8XKC2 56662962 IC50 > 100000 nM T04831 C0T8QZ 56662963 IC50 = 100 nM T04831 COH9G3 56666393 IC50 = 48000 nM T04831 CJD0P8 56666438 IC50 > 100000 nM T04831 C36XYF 56666439 IC50 = 18000 nM T04831 CA42FJ 56666467 IC50 = 11000 nM T04831 C3JT6B 56669804 IC50 = 300 nM T04831 C6X5UV 56669805 IC50 = 8000 nM T04831 C1Q8AD 56669806 IC50 = 100 nM T04831 CG1IT9 56669852 IC50 = 1500 nM T04831 CND1T2 56669853 IC50 = 50000 nM T04831 CM5FL6 56673297 IC50 = 55000 nM T04831 CA32UJ 56673389 IC50 = 14000 nM T04831 C87RUH 56673390 IC50 = 12000 nM T04831 CET8S0 56676623 IC50 = 19000 nM T04831 CM40ON 56676624 IC50 = 51000 nM T04831 CHR3M8 56676675 IC50 > 100000 nM T04831 C30BIC 56676676 IC50 = 45000 nM T04831 CEZ39Y 56679958 IC50 = 3500 nM T04831 CW04DN 56679959 IC50 = 2500 nM T04831 CDEM30 56679960 IC50 = 7000 nM T04831 CB1H6Z 56679961 IC50 > 100000 nM T04831 CH1UK6 56680023 IC50 = 750 nM T04831 C5KB4E 56680024 IC50 = 11000 nM T04831 CS1U2A 56683286 IC50 > 100000 nM T04831 CGX39M 56683287 IC50 = 150 nM T04831 CUO35I 56683288 IC50 = 50000 nM T04831 CKF34Z 56683289 IC50 > 100000 nM T04831 C3P0FG 56683334 IC50 > 100000 nM T04831 CX4H6I 86583042 IC50 > 10000 nM T04831 C4TXF2 118730409 IC50 = 480000 nM T04831 CW3OF5 135398511 IC50 < 100 nM T04831 C5L7IE 135411750 IC50 = 10500 nM T04831 C5RNG3 135432788 IC50 = 4000 nM T04831 C2D5WG 135653128 IC50 = 3000 nM T04831 CXC69T 137321158 IC50 = 210 nM T04831 C2MD1Q 155513187 IC50 > 10000 nM T04831 D02PVB 8515 IC50 = 8000 nM T04831 D04WFN 10202471 IC50 = 2000 nM T04831 D06KDU 16760346 IC50 = 7000 nM T04831 D06KSF 9549300 IC50 = 250 nM T04831 D07OCA 5330812 IC50 = 1600 nM T04831 D09RES 11665831 IC50 = 12000 nM T04831 D0A7FQ 11644425 IC50 = 5000 nM T04831 D0D2FC 2794188 IC50 = 3000 nM T04831 D0D5HQ 5330797 IC50 = 6000 nM T04831 D0E0XV 9903786 IC50 = 250 nM T04831 D0HZ8U 3467590 IC50 < 100 nM T04831 D0L3FK 5289419 IC50 = 5000 nM T04831 D0N4LR 53469448 IC50 = 696 nM T04831 D0Q3EW 9549303 IC50 = 20000 nM T04831 D0Q7TO 6419766 IC50 = 15000 nM T04831 D0R5FH 438981 IC50 = 6000 nM T04831 D0T8KR 9549289 IC50 = 4000 nM T04831 D0Y0BK 11524144 IC50 = 16000 nM T04831 D0Y0ES 3707 IC50 < 100 nM T04831 D0Z2CN 135418335 IC50 < 100 nM T04902 CYNF54 114619 IC50 = 104 nM T04902 C3YF4P 462382 Ki = 653 nM T04902 CK4X9E 5353866 Ki = 5330 nM T04902 C8W9ER 9827472 Ki = 41 nM T04902 CZ3MO5 9839500 Ki = 370 nM T04902 COAM65 9844151 Ki = 5 nM T04902 CYAC30 9910792 Ki = 180 nM T04902 CF5W3H 9984343 Ki = 17 nM T04902 CN18SE 10456222 IC50 = 184 nM T04902 CN8PB5 10649378 Ki = 5 nM T04902 C3VCM6 10690823 Ki = 13 nM T04902 C0XE7T 10740734 Ki = 9 nM T04902 C5SN8Q 10786038 Ki = 11 nM T04902 CD72KH 10788273 Ki = 7 nM T04902 CN0F8E 11199915 IC50 = 350 nM T04902 C3OI2T 15017709 IC50 = 104 nM T04902 CUA19Y 16760339 Ki = 210 nM T04902 CYA5V6 16760340 Ki = 120 nM T04902 C2GXK0 23240732 Ki = 400 nM T04902 C52GAL 23240733 Ki = 400 nM T04902 CT6PW7 23240734 Ki = 19 nM T04902 CJD86W 23240735 Ki = 44 nM T04902 C5SX7Z 23240736 Ki = 19 nM T04902 C6YW0C 23240737 Ki = 22 nM T04902 C15TFI 23240738 Ki = 39 nM T04902 C2NRA7 23240739 Ki = 24 nM T04902 C5UQT7 23240740 Ki = 5.7 nM T04902 CI89XA 23240741 Ki = 22 nM T04902 CB98KA 24771859 IC50 = 30 nM T04902 CDO07M 25231938 IC50 = 850 nM T04902 C9NI1O 25231939 IC50 = 1100 nM T04902 CJB3L1 25231940 IC50 = 28000 nM T04902 CA1Z2M 25232114 IC50 = 31000 nM T04902 CHV5W6 25232115 IC50 = 700 nM T04902 C1E8PY 25232116 IC50 = 180 nM T04902 CZN61Q 25232117 IC50 = 1010 nM T04902 C5FY9H 44284219 IC50 = 184 nM T04902 CT4FH7 44284304 IC50 = 79.6 nM T04902 C5OT0F 44323240 Ki = 7 nM T04902 CMX96T 44330903 Ki = 42 nM T04902 CUM39I 44330915 Ki = 35 nM T04902 CPNJ80 44330944 Ki = 122 nM T04902 CAEG80 44343472 Ki = 400 nM T04902 C1IPZ6 44343473 Ki = 1500 nM T04902 CN5GQ3 44343531 Ki = 50 nM T04902 C15XLB 44343546 Ki = 59 nM T04902 CB53OZ 44343547 Ki = 760 nM T04902 C02RUT 44343554 Ki = 1600 nM T04902 C1WM7R 44343562 Ki = 63 nM T04902 CGN37W 44343594 Ki = 43 nM T04902 C47KQO 44343612 Ki = 22 nM T04902 C6E9HW 44343648 Ki = 250 nM T04902 C6J1WX 44343650 Ki = 600 nM T04902 C3V5XU 44343661 Ki = 200 nM T04902 CVR40J 44343678 Ki = 1200 nM T04902 C4G1DX 44343691 Ki = 78 nM T04902 C7LH3U 44343713 Ki = 1200 nM T04902 CU4DC6 44343744 Ki = 28 nM T04902 CW2Z7I 44343748 Ki = 46 nM T04902 C8SFT5 44343749 Ki = 65 nM T04902 C7L2RA 44343763 Ki = 88 nM T04902 C78DRG 44343802 Ki = 17000 nM T04902 CYIN64 44343847 Ki = 500 nM T04902 C0OSC3 44343848 Ki = 470 nM T04902 CNO65Y 44343910 Ki = 140 nM T04902 C17NVX 44343911 Ki = 50 nM T04902 CJK58F 44343915 Ki = 2900 nM T04902 CVKL43 44343918 Ki = 67 nM T04902 CX3OJ2 44343945 Ki = 1600 nM T04902 CUE8J0 44343946 Ki = 1900 nM T04902 CN4XE3 44343970 Ki = 2200 nM T04902 CFR7P1 44343971 Ki = 1400 nM T04902 CE7YB4 44344038 Ki = 1100 nM T04902 CSWU72 44344051 Ki = 400 nM T04902 C6X9JO 44353497 Ki = 110 nM T04902 CVHL49 44353498 Ki = 300 nM T04902 C50JMZ 44353509 Ki = 9900 nM T04902 C1R7HO 44353510 Ki = 480 nM T04902 CD1KB5 44353514 Ki = 11000 nM T04902 CT43EV 44353526 Ki = 580 nM T04902 CV6U1K 44353527 Ki = 100 nM T04902 CN15EA 44353530 Ki = 83 nM T04902 CKH5Y4 44353532 Ki = 290 nM T04902 CK35CO 44353533 Ki = 350 nM T04902 CUFZ01 44353534 Ki = 310 nM T04902 CN6B8M 44353535 Ki = 50 nM T04902 C0T4MF 44353540 Ki = 830 nM T04902 CP5NY3 44353544 Ki = 76 nM T04902 CB1HC7 44353545 Ki = 200 nM T04902 C5FXE6 44353552 Ki = 68 nM T04902 CH3BQ1 44353553 Ki = 1200 nM T04902 CJ0Y3M 44353556 Ki = 160 nM T04902 C1QG3Z 44353580 Ki = 46 nM T04902 C6T3DA 44353581 Ki = 86 nM T04902 CV6U5Q 44353582 Ki = 160 nM T04902 CMTJ91 44353589 Ki = 250 nM T04902 CM3R5T 44353590 Ki = 160 nM T04902 CZ2YG8 44353593 Ki = 470 nM T04902 CY6CK7 44353594 Ki = 120 nM T04902 CFZ36E 44353603 Ki = 160 nM T04902 C6MV2C 44353604 Ki = 330 nM T04902 CWV2C8 44353606 Ki = 160 nM T04902 CEJ3D8 44353608 Ki = 110 nM T04902 C8YPO1 44353613 Ki = 60 nM T04902 C0WIP1 44353630 Ki = 360 nM T04902 CT3Q8G 44353631 Ki = 730 nM T04902 C6BQS9 44353632 Ki = 110 nM T04902 C7DRX0 44353633 Ki = 90 nM T04902 C0T5HM 44353640 Ki = 130 nM T04902 CS9VG4 44353649 Ki = 78 nM T04902 CI9UB0 44353680 Ki = 100 nM T04902 C1V8RS 44353769 Ki = 17 nM T04902 C53QGD 44353782 Ki = 66 nM T04902 C91OHB 44353783 Ki = 33 nM T04902 CUY2N7 44353792 Ki = 270 nM T04902 C5XVK9 44353793 Ki = 22 nM T04902 CTD5O8 44353799 Ki = 150 nM T04902 CH80QO 44353801 Ki = 69 nM T04902 CNM2U3 44353805 Ki = 280 nM T04902 CF8ZU0 44353806 Ki = 4600 nM T04902 CV97ZN 44353808 Ki = 290 nM T04902 CG6Q3F 44353809 Ki = 590 nM T04902 C8O3LK 44353810 Ki = 180 nM T04902 CMP1Z0 44353811 Ki = 200 nM T04902 CPA90D 44353812 Ki = 150 nM T04902 C49MCW 44353814 Ki = 600 nM T04902 CN9W5C 44353816 Ki = 240 nM T04902 CX3RZ0 44353817 Ki = 170 nM T04902 CCEU50 44353818 Ki = 100 nM T04902 C57SFJ 44353819 Ki = 670 nM T04902 CX9LJ0 44353820 Ki = 120 nM T04902 C9PY1J 44353821 Ki = 450 nM T04902 CU74GM 44353822 Ki = 110 nM T04902 CDHX90 44353823 Ki = 170 nM T04902 CQ9BT7 44353833 Ki = 410 nM T04902 CT21FG 44353834 Ki = 220 nM T04902 CZ3XP9 44353836 Ki = 50 nM T04902 CB7I6Q 44353838 Ki = 340 nM T04902 CB7P0H 44353839 Ki = 74 nM T04902 CF3A0M 44353840 Ki = 280 nM T04902 CS5DX4 44353841 Ki = 120 nM T04902 CZ89JO 44353846 Ki = 51 nM T04902 CP3VT2 44353858 Ki = 270 nM T04902 C5H9VR 44353859 Ki = 23 nM T04902 C1HR8U 44353865 Ki = 120 nM T04902 CE5V7Y 57390763 IC50 = 85 nM T04902 C9T3JY 57391494 IC50 = 2400 nM T04902 CHK83B 57391503 IC50 = 3710 nM T04902 CLX4Q5 57394298 IC50 = 295 nM T04902 C3NXM9 57394973 IC50 = 280 nM T04902 C8ITL0 73107490 Ki = 190 nM T04902 C2Y6TO 73347008 Ki = 2600 nM T04902 CTA8U5 85090477 Ki = 200 nM T04902 CC2LB9 90663209 Ki = 1900 nM T04902 C4ZH1J 90663211 Ki = 260 nM T04902 CQ42NT 90663212 Ki = 1400 nM T04902 C52LCE 90663213 Ki = 90 nM T04902 CGQ18K 122197351 Ki = 200 nM T04902 CX7FP8 122197352 Ki = 260 nM T04902 CXM6Z0 127051056 Ki = 2028 nM T04902 CJ7O6G 127051057 Ki = 2983 nM T04902 C6B2ZU 127051058 Ki = 1708 nM T04902 D03UYO 44353781 Ki = 15 nM T81658 D05VZE 119031 IC50 = 10000 nM T81658 D0T9HG 132519 IC50 = 6 nM T81658 CJS23I 9868333 Ki > 7088 nM T81658 CG38KL 9936728 Ki = 71 nM T81658 CR7T3J 10009978 Ki > 2000 nM T81658 CR5H6E 10163627 Ki > 7088 nM T81658 CK0P3F 10186536 Ki > 7088 nM T81658 C4K1MJ 10208262 Ki > 7088 nM T81658 CY08WJ 10322755 Ki = 1700 nM T81658 C6WZ4F 10367355 IC50 = 4 nM T81658 CFKA79 10395015 Ki > 2000 nM T81658 C5WV1N 10439082 Ki > 2000 nM T81658 C8C5AV 11294179 Ki > 10000 nM T81658 CO8QT0 11753905 Ki > 7100 nM T81658 C02BWA 11967143 Ki > 2000 nM T81658 C75XDI 16730519 IC50 > 7000 nM T81658 CAQ9Z1 25022681 Ki > 7088 nM T81658 CHR2P1 25183768 Ki > 25000 nM T81658 CGQ92A 44364037 IC50 = 44 nM T81658 C36YLM 44364111 IC50 = 385 nM T81658 CN4T7Q 44364119 IC50 = 126 nM T81658 CH4TE7 44364121 IC50 = 17 nM T81658 CPE91Y 44364122 IC50 = 19 nM T81658 CG2X0C 44364224 IC50 = 218 nM T81658 C1F8XN 44364249 IC50 = 6 nM T81658 CWM47H 44364250 IC50 = 29 nM T81658 C0W5TL 44364251 IC50 = 7303 nM T81658 C3TPO7 44364266 IC50 = 1789 nM T81658 CJ2B8F 44364280 IC50 = 621 nM T81658 CK68GT 44580539 IC50 > 5000 nM T81658 CU2SX3 51355576 Ki > 10000 nM T81658 D07GEL 10344307 Ki = 20 nM T81658 D0H6CK 10160968 Ki > 7088 nM T81658 D0L4EO 11609208 IC50 = 13940 nM T81658 D0W2UK 6914621 Ki = 3997 nM T59328 D01PZD 5329098 IC50 > 100000 nM T59328 D03MNN 11341869 IC50 = 230 nM T59328 D03ZBT 11626560 IC50 = 681 nM T59328 D04LVK 57379345 IC50 = 28 nM T59328 D05NUH 54758501 IC50 = 10 nM T59328 D05UFG 10184653 IC50 = 0.19 nM T59328 D06IAR 60961 IC50 = 195000 nM T59328 D06XXH 11511120 IC50 = 1.8 nM T59328 D07POC 176870 Ki = 0.1 nM T59328 D08CDI 208908 Ki = 3 nM T59328 D08HVR 6047 IC50 = 900000 nM T59328 D08PIE 68165256 IC50 = 1 nM T59328 D09KTS 24821094 IC50 = 0.75 nM T59328 D09PQZ 71226662 IC50 > 2000 nM T59328 D09XZB 123631 IC50 = 0.1 nM T59328 D0AZ3C 5291 IC50 > 100000 nM T59328 D0B0AX 5328127 IC50 = 50000 nM T59328 D0C4RB 36314 IC50 > 10000 nM T59328 D0E6XR 3062316 IC50 = 180 nM T59328 D0EG1I 9926791 IC50 > 10000 nM T59328 D0G6QF 3081361 IC50 = 200 nM T59328 D0GY5Z 2244 IC50 > 10000 nM T59328 D0H0EQ 24826799 IC50 > 1000 nM T59328 D0IQ6P 25102847 IC50 = 19 nM T59328 D0J9ZR 4477 IC50 = 10500 nM T59328 D0K8KX 5280343 IC50 = 900 nM T59328 D0O8GK 71496458 IC50 = 0.421 nM T59328 D0OB0F 5328940 IC50 = 53 nM T59328 D0R0MW 5329102 IC50 = 140 nM T59328 D0R1QE 3672 IC50 > 10000 nM T59328 D0R1RS 3715 IC50 > 10000 nM T59328 D0W5HK 216239 IC50 = 43.5 nM T59328 D0W9WF 3825 IC50 > 10000 nM T59328 D0Y9EW 42611257 IC50 > 10000 nM T59328 D0Z5IU 1548887 IC50 > 10000 nM T59328 D00NYJ 42642648 IC50 = 7 nM T59328 D00RMC 6918508 IC50 = 3 nM T59328 D00YER 25127713 IC50 = 0.218 nM T59328 D01GFX 11640390 IC50 > 12500 nM T59328 D02BYZ 71667668 IC50 = 8 nM T59328 D02RJY 11442891 IC50 > 10000 nM T59328 D02TUL 118115473 IC50 > 50000 nM T59328 D02UFQ 11620908 IC50 = 1 nM T59328 D03LWG 53235510 IC50 > 10000 nM T59328 D04BFC 59174488 IC50 = 442 nM T59328 D06WRF 10458325 IC50 = 0.3 nM T59328 D07EHV 44814409 IC50 > 10000 nM T59328 D07HPJ 11476171 IC50 = 5200 nM T59328 D09TAB 25151352 IC50 > 10000 nM T59328 D0A1AQ 5329099 IC50 > 100000 nM T59328 D0BM7M 11488320 IC50 = 4 nM T59328 D0CN9Q 9874913 IC50 = 6400 nM T59328 D0D1GF 42642645 IC50 = 2990 nM T59328 D0E3TC 44259 IC50 = 0.38 nM T59328 D0G2QH 10297043 IC50 = 2 nM T59328 D0G5XV 135565884 IC50 = 2.6 nM T59328 D0HS5V 11234052 IC50 > 1900 nM T59328 D0I1DW 9808998 IC50 > 200000 nM T59328 D0K7FY 72703790 IC50 = 160.6 nM T59328 D0L4FS 5280961 IC50 = 0.1 ug.mL-1 T59328 D0LF1U 5287969 IC50 = 7600 nM T59328 D0M0XB 10302451 IC50 = 66 nM T59328 D0M4AV 57335384 IC50 = 1.6 nM T59328 D0O0LS 25141092 IC50 > 10000 nM T59328 D0O6WV 24794418 IC50 > 12500 nM T59328 D0P1CV 46191454 IC50 > 10000 nM T59328 D0P6DJ 151194 IC50 = 457.7 nM T59328 D0Q7RE 16007391 Ki > 10000 nM T59328 D0Q9CY 9915743 IC50 = 0.08 nM T59328 D0Q9UX 16718576 IC50 = 3069 nM T59328 D0QX8X 71479709 IC50 = 5800 nM T59328 D0R0LB 91668194 IC50 = 12 nM T59328 D0S3PO 6445562 IC50 = 8.02 nM T59328 D0S5RC 3025986 IC50 > 25000 nM T59328 D0U4FF 10437018 IC50 = 32 nM T59328 D0VF6E 1401 IC50 > 50000 nM T59328 D0X4MN 11597537 IC50 = 380 nM T59328 D0YB3W 156414 Ki = 0.11 nM T59328 D0Z4RC 24756910 IC50 = 2.4 nM T59328 D0ZN1R 68245 IC50 = 6.27 nM T59328 D03BNU 59604787 IC50 > 3500 nM T59328 D0LF0O 135441202 IC50 = 21000 nM T59328 D04SWX 56924694 IC50 = 113 nM T59328 D0NH9P 135 IC50 = 10 ug.mL-1 T59328 D0OE4F 4369496 IC50 > 100000 nM T59328 D00BPA 4592 IC50 = 440000 nM T59328 D01EFO 9864718 IC50 = 65000 nM T59328 D02YAQ 6603857 IC50 = 1 nM T59328 D03QTP 1697 Ki = 160 nM T59328 D03WTT 5468216 IC50 = 700 nM T59328 D04FHB 6918852 Ki > 5000 nM T59328 D07GFF 6918403 IC50 = 3.7 nM T59328 D08DBE 10344820 Ki = 35 nM T59328 D0A9KI 9863367 IC50 > 10 nM T59328 D0B3CT 9928668 IC50 = 29000 nM T59328 D0D5CJ 9818362 IC50 > 100000 nM T59328 D0F8DL 176155 IC50 > 33000 nM T59328 D0GZ7B 5328779 IC50 = 501.19 nM T59328 D0H8KG 5311382 IC50 = 44000 nM T59328 D0HO1S 6711154 IC50 = 700 nM T59328 D0IT6Q 3038522 IC50 > 30000 nM T59328 D0L5YF 5329032 IC50 = 50 nM T59328 D0Q7HO 4705 Ki = 0.006 nM T59328 D0T3ME 156422 IC50 = 3800 nM T59328 C0U5TZ 1302 IC50 > 10000 nM T59328 CB1VW3 1400 Ki = 199.53 nM T59328 C03TMS 1714 IC50 = 126.7 nM T59328 CO8C3E 2046 Ki = 150000 nM T59328 CH21PG 2428 IC50 = 0.008 nM T59328 C8HN2C 3798 IC50 = 29 nM T59328 C1BE5N 3799 IC50 = 10000 nM T59328 C2LS4F 3895 IC50 = 0.5 ug.mL-1 T59328 C0W4UD 3896 IC50 = 30 nM T59328 C2DUS8 4706 IC50 = 0.69 nM T59328 CBPM40 4878 IC50 = 480 nM T59328 CKZH57 5613 IC50 = 6500000 nM T59328 C2I3WC 5614 Ki = 155000 nM T59328 CQAO39 9210 IC50 = 27 nM T59328 CO7NY6 18091 Ki = 117000 nM T59328 C8K2FU 18606 IC50 > 1250000 nM T59328 CN31AP 19424 Ki = 67000 nM T59328 C12BXO 23905 IC50 = 225000 nM T59328 CL3H9Z 33296 IC50 > 325000 nM T59328 C0TMU5 37583 IC50 = 1400000 nM T59328 C4D5OH 44390 IC50 = 250000 nM T59328 C43WLX 57591 Ki = 50000 nM T59328 C62EPW 58857 Ki = 55000 nM T59328 CQD56Z 73299 IC50 > 20000 nM T59328 C63WLY 89644 IC50 = 6 ug.mL-1 T59328 CE4K5D 92516 IC50 > 50000 nM T59328 CI27WO 92970 Ki = 160000 nM T59328 C5JE2Z 104860 IC50 = 3.5 ug.mL-1 T59328 CF5B3H 121059 IC50 = 600000 nM T59328 C91ERH 128872 IC50 = 23 nM T59328 C6Y9CV 151193 IC50 > 10000 nM T59328 CRFU83 156413 IC50 = 1.5 nM T59328 CA5CO8 157820 IC50 > 100000 nM T59328 CI1NA5 159926 IC50 = 2.7 ug.mL-1 T59328 CI80NA 160436 IC50 > 50000 nM T59328 CV7W4J 176406 IC50 = 2511.89 nM T59328 C2P8XO 176871 IC50 = 70 nM T59328 CYBA43 177458 IC50 = 4 ug.mL-1 T59328 CPI83T 198909 IC50 = 4100 nM T59328 CRP4A8 244537 IC50 > 250000 nM T59328 C8MUX3 252473 Ki = 123000 nM T59328 C4C7HJ 282723 Ki > 400000 nM T59328 C61DPM 321779 Ki > 250000 nM T59328 CPF26C 324081 IC50 = 344 nM T59328 C9WA8F 341040 IC50 = 5600 nM T59328 CL1M8I 350716 IC50 > 50000 nM T59328 CV3XI1 354479 IC50 = 350 nM T59328 CZ5B0Y 367524 Ki > 400000 nM T59328 C0DI9H 375472 IC50 = 5000 nM T59328 C0M4OG 375473 IC50 = 3300 nM T59328 CMH0V9 382059 IC50 = 10 nM T59328 CQX5W6 390508 IC50 = 10000 nM T59328 CPF67R 402810 IC50 = 41900 nM T59328 CNP3M1 403661 IC50 = 320000 nM T59328 CC2R6G 409975 IC50 = 1800 nM T59328 CK0L4O 442514 IC50 = 3400 nM T59328 C4MNG8 445840 IC50 > 20000 nM T59328 C1YNB7 447721 IC50 > 10000 nM T59328 C1ZG2U 449087 IC50 > 10000 nM T59328 CT5O9L 519420 IC50 = 1500000 nM T59328 CSA52V 542795 IC50 > 20000 nM T59328 CVQ2Y4 589288 IC50 = 0.79 nM T59328 CO0U5E 616443 IC50 > 20000 nM T59328 C53PTU 616573 IC50 = 320 nM T59328 C2U6LB 643159 IC50 = 850000 nM T59328 C75EDQ 644355 IC50 > 30000 nM T59328 C5HPF3 644356 IC50 > 30000 nM T59328 CSA18D 651672 IC50 = 577 nM T59328 CJ0YU6 659954 IC50 = 912.01 nM T59328 CR3N8A 667645 Ki = 2200 nM T59328 CP91NX 677915 IC50 = 14590 nM T59328 CLEU84 689033 IC50 > 100000 nM T59328 CDE9V2 689424 IC50 = 19690 nM T59328 C5O0TJ 690158 IC50 = 23160 nM T59328 C7TPR6 690965 IC50 = 9050 nM T59328 C3Q6IY 694087 IC50 > 100000 nM T59328 C3V5KD 694921 IC50 > 250000 nM T59328 CX17CH 701322 IC50 = 63 nM T59328 C34EXB 702486 IC50 = 13930 nM T59328 CYO86G 703960 IC50 > 100000 nM T59328 C4BX6T 707914 IC50 = 560000 nM T59328 CD69IF 710163 IC50 > 625000 nM T59328 C65SGT 712193 IC50 = 842 nM T59328 C6D4HT 720879 IC50 = 325000 nM T59328 C6CJY8 725409 IC50 = 30 nM T59328 CTO15S 727131 IC50 = 10020 nM T59328 C9D7UY 727518 IC50 > 100000 nM T59328 C2CL6X 732134 IC50 = 5160 nM T59328 CKO38Q 732136 IC50 = 10230 nM T59328 C6AKG9 735124 IC50 = 56 nM T59328 C17UDE 735126 IC50 = 80 nM T59328 C4V7OW 736236 IC50 = 833000 nM T59328 CT7E1K 746495 Ki = 300000 nM T59328 C6ECP2 755464 IC50 = 11690 nM T59328 CWZY50 764334 IC50 = 15740 nM T59328 CPKI76 765318 IC50 = 9860 nM T59328 CXME85 766168 IC50 = 13710 nM T59328 CB30XT 778859 IC50 = 16170 nM T59328 CQB03J 780790 IC50 = 12290 nM T59328 C7EHR1 787183 IC50 = 12690 nM T59328 CLU06E 792233 IC50 = 14580 nM T59328 C73TME 811665 IC50 = 12320 nM T59328 CTX13N 814517 IC50 = 460 nM T59328 CB27WS 849733 IC50 > 10000 nM T59328 CW56XG 875024 IC50 = 7370 nM T59328 CP40SX 889945 IC50 = 5720 nM T59328 C5GMN8 935994 IC50 = 149 nM T59328 CXB5A2 964113 IC50 > 100000 nM T59328 CW7FM4 967629 IC50 = 26060 nM T59328 C7SD1U 1007600 IC50 = 3500 nM T59328 C9DBI2 1011523 IC50 = 9700 nM T59328 C0NF2R 1018252 IC50 = 5600 nM T59328 CR8F6B 1035343 IC50 > 100000 nM T59328 CEF7B3 1086535 IC50 = 8400 nM T59328 C9U7NK 1128774 IC50 = 76700 nM T59328 CQWX85 1304420 IC50 = 15000 nM T59328 CJP04L 1474852 IC50 = 0.07244 nM T59328 CYQ90E 1474874 IC50 > 1000 nM T59328 C6OC3G 1474877 IC50 = 10 nM T59328 CC3A8B 1474883 IC50 = 3.8 nM T59328 CK3QN1 1475063 IC50 = 19.1 nM T59328 C3SGW1 1490236 IC50 = 3000 nM T59328 CMYK57 1500232 IC50 = 24830 nM T59328 C84MXV 1500233 IC50 > 30000 nM T59328 CDB17F 1538822 IC50 = 18500 nM T59328 CG73KY 1550166 Ki = 1400000 nM T59328 C2BCN0 1550170 IC50 = 833000 nM T59328 CRQ82G 1558661 Ki = 1350000 nM T59328 CSA69X 1637668 IC50 = 9350 nM T59328 C6ZY1V 1641261 IC50 > 20000 nM T59328 C5WM1Q 1723871 IC50 = 8600 nM T59328 CL6IN7 1742852 IC50 = 74300 nM T59328 CVA45M 1810492 IC50 = 23100 nM T59328 C1P4FC 1838043 IC50 = 12022.64 nM T59328 CDC7Q4 1900460 IC50 = 35800 nM T59328 C71YPT 2103474 IC50 = 35 nM T59328 CZ2B4M 2358462 IC50 > 100000 nM T59328 CXA1L7 2365265 IC50 > 100000 nM T59328 CEF62M 2379240 IC50 > 100000 nM T59328 CS6RH2 2385464 IC50 = 5888.44 nM T59328 C7EB0A 2385467 IC50 = 2000 nM T59328 CKT64G 2396126 IC50 > 10000 nM T59328 C6T0OJ 2400783 IC50 = 2980 nM T59328 CKE7P2 2725645 IC50 = 200 nM T59328 C31KAP 2743369 IC50 = 54 nM T59328 C5ON0G 2744121 IC50 > 100000 nM T59328 C9IWU0 2789324 IC50 = 50 nM T59328 C4POJ7 2795373 IC50 = 260000 nM T59328 CG43CZ 2802451 IC50 = 2520 nM T59328 C8S0UP 2806990 IC50 = 45500 nM T59328 CV7Y5T 2807058 IC50 = 1500 nM T59328 C8VD6N 2808930 IC50 > 3240 nM T59328 C0KB3P 2810857 IC50 = 11100 nM T59328 CEX1W9 2811342 IC50 > 100000 nM T59328 CSA5I6 2839887 IC50 = 6270 nM T59328 C9VUX8 2843335 IC50 = 16630 nM T59328 C3BJP7 2943601 IC50 > 10000 nM T59328 C8HAL7 2983225 IC50 = 38430 nM T59328 CFVK40 3008950 IC50 > 50000 nM T59328 CD8UW1 3008956 IC50 = 200 nM T59328 CCD93P 3008957 IC50 = 1240 nM T59328 CU64VM 3008958 IC50 = 1670 nM T59328 C8F0KM 3008959 IC50 = 4310 nM T59328 CV8R9Z 3008960 IC50 = 6160 nM T59328 C8EZ6O 3008961 IC50 = 9190 nM T59328 CX95SU 3008962 IC50 = 12620 nM T59328 C9B2MN 3008963 IC50 = 17420 nM T59328 C9E7BW 3008964 IC50 = 19770 nM T59328 CGK91Q 3008965 IC50 > 50000 nM T59328 CHGP54 3035187 IC50 = 0.8 nM T59328 CJBX04 3039851 IC50 = 1500 nM T59328 CHK3W2 3135836 IC50 = 92400 nM T59328 C2SM4G 3138425 IC50 = 81600 nM T59328 CCN9D5 3142817 IC50 = 280 nM T59328 CUK5Y1 3374314 IC50 = 20000 nM T59328 CW74LV 3564138 IC50 > 10000 nM T59328 C3QSK2 3677514 IC50 = 72400 nM T59328 C46IJS 3724145 IC50 = 5110 nM T59328 CCUW85 4205046 IC50 = 4300 nM T59328 CPHI06 4321095 IC50 > 100000 nM T59328 CZB15R 4350438 IC50 = 2000 nM T59328 CM5VN6 4600415 IC50 = 88670 nM T59328 C8O9MN 4616059 IC50 = 1330 nM T59328 C2W4OD 4677622 IC50 = 20190 nM T59328 CN7MT6 4750207 IC50 = 31000 nM T59328 CB3G6R 4913175 IC50 = 200 nM T59328 CSI43N 5083839 IC50 = 28690 nM T59328 C1BPI8 5280569 IC50 = 7670 nM T59328 C8N6AY 5281377 IC50 > 100 ug.mL-1 T59328 C4JB3P 5281801 IC50 = 3 ug.mL-1 T59328 C0FLB1 5281811 IC50 = 3300 nM T59328 CTID76 5282335 IC50 > 25000 nM T59328 CY28LS 5293755 IC50 > 100000 nM T59328 CW26CH 5311106 IC50 > 20000 nM T59328 C4VTS3 5327723 IC50 > 100000 nM T59328 C6UL3A 5327821 IC50 = 220 nM T59328 CR3OF4 5327822 IC50 = 160 nM T59328 C9QMX2 5327823 IC50 = 58 nM T59328 CA4G1B 5327824 IC50 = 84 nM T59328 CY2NC3 5327825 IC50 = 250 nM T59328 CDT07K 5327826 IC50 < 800 nM T59328 CG36XB 5327827 IC50 = 130 nM T59328 CF3Y6G 5327828 IC50 = 30 nM T59328 CY1Z9E 5327829 IC50 = 8 nM T59328 CI51CH 5327830 IC50 = 8 nM T59328 CUAW78 5327831 IC50 = 4 nM T59328 CC9US2 5327832 IC50 > 100000 nM T59328 CVGK98 5327833 IC50 = 5 nM T59328 CGWP86 5327834 IC50 = 29 nM T59328 C10RVD 5327835 IC50 = 3 nM T59328 CD6B2A 5327836 IC50 = 26 nM T59328 CY1O6K 5327837 IC50 = 8 nM T59328 C1K8CJ 5327838 IC50 = 7 nM T59328 CP15JO 5327839 IC50 = 19 nM T59328 CWT9S8 5327840 IC50 = 26 nM T59328 C5EWD2 5327841 IC50 = 96 nM T59328 C67JVQ 5327843 IC50 = 270 nM T59328 CY23QP 5327844 IC50 = 5 nM T59328 CN1X4Z 5327845 IC50 = 270 nM T59328 C6TGI1 5327846 IC50 = 2 nM T59328 CEMR07 5327847 IC50 = 24200 nM T59328 CB90GI 5327848 IC50 = 1500 nM T59328 CMC76E 5327864 IC50 = 5600 nM T59328 C43JFT 5327866 IC50 > 50000 nM T59328 C4ZW0Q 5327868 IC50 = 7500 nM T59328 CY82TU 5327869 IC50 = 4500 nM T59328 CL4OG5 5327870 IC50 > 5000 nM T59328 CYGA64 5327871 IC50 = 4400 nM T59328 CZE87D 5327872 IC50 > 50000 nM T59328 C7XOK5 5327873 IC50 > 5000 nM T59328 CQK5Z0 5327874 IC50 > 50000 nM T59328 CS0Q4N 5327875 IC50 > 50000 nM T59328 CI96EG 5327876 IC50 = 1400 nM T59328 CT86OE 5327877 IC50 > 5000 nM T59328 C23EZX 5327878 IC50 = 8700 nM T59328 C63SAG 5327879 IC50 = 210 nM T59328 CT94BD 5327880 IC50 = 4500 nM T59328 CNRS28 5327881 IC50 > 5000 nM T59328 CD43FT 5327882 IC50 > 5000 nM T59328 CX39AM 5327883 IC50 > 5000 nM T59328 CZWG61 5327884 IC50 = 1000 nM T59328 C3P8CG 5327885 IC50 = 260 nM T59328 CWZ8H3 5327886 IC50 = 200 nM T59328 CC7VR3 5327887 IC50 = 510 nM T59328 CG7Q3R 5327888 IC50 = 1300 nM T59328 CYRW80 5327889 IC50 = 910 nM T59328 C7W8IJ 5327890 IC50 = 490 nM T59328 CJ28SO 5327891 IC50 > 5000 nM T59328 C82PDN 5327892 IC50 = 670 nM T59328 C52MYD 5327893 IC50 = 480 nM T59328 C4ET5H 5327894 IC50 = 66 nM T59328 CJ5VO8 5327895 IC50 = 30 nM T59328 CDA78E 5327896 IC50 = 220 nM T59328 CQ0ZP3 5327897 IC50 = 150 nM T59328 COQH79 5327899 IC50 = 250 nM T59328 C9R8DP 5327900 IC50 = 330 nM T59328 CVB9L3 5327902 IC50 > 50000 nM T59328 C7EK0Z 5327903 IC50 = 700 nM T59328 CN71AK 5327916 IC50 = 190 nM T59328 C5JI1A 5327917 IC50 = 220 nM T59328 C4CWI1 5327918 IC50 = 80 nM T59328 CQ0J3U 5328014 IC50 = 7000 nM T59328 C0FCR1 5328015 IC50 = 10000 nM T59328 C5VW6K 5328016 IC50 > 50000 nM T59328 C5IL6F 5328017 IC50 > 1000 nM T59328 C6RHB3 5328018 IC50 = 756 nM T59328 C5FXG1 5328019 IC50 = 5500 nM T59328 CPF5M1 5328020 IC50 > 10000 nM T59328 CKOI31 5328021 IC50 > 100000 nM T59328 CV5IX3 5328022 IC50 > 100000 nM T59328 CK31WA 5328023 IC50 > 1000 nM T59328 CFH4N1 5328024 IC50 = 8000 nM T59328 C89PLV 5328025 IC50 > 10000 nM T59328 CWE6K5 5328026 IC50 = 4900 nM T59328 CH5R7E 5328027 IC50 > 10000 nM T59328 CU6F0M 5328028 IC50 = 508 nM T59328 C0N4ZK 5328029 IC50 = 200 nM T59328 CYVQ61 5328030 IC50 = 5900 nM T59328 CP4AW6 5328031 IC50 > 1000 nM T59328 CH0J3D 5328032 IC50 = 58 nM T59328 C6R2HK 5328033 IC50 > 10000 nM T59328 CG2PT3 5328034 IC50 > 10000 nM T59328 C8BEX5 5328035 IC50 > 10000 nM T59328 C7KO4J 5328037 IC50 = 56 nM T59328 C7NAH0 5328039 IC50 = 439 nM T59328 CIRD30 5328040 IC50 = 139 nM T59328 CCL34N 5328041 IC50 = 897 nM T59328 C0SF3M 5328043 IC50 = 30 nM T59328 C8N1PH 5328044 IC50 = 1000 nM T59328 CCZP83 5328046 IC50 = 10 nM T59328 CG94OR 5328047 IC50 > 10000 nM T59328 C1AEK5 5328048 IC50 = 105 nM T59328 C0W1KQ 5328049 IC50 = 974 nM T59328 C5VS7Z 5328051 IC50 = 250 nM T59328 C8MK4H 5328052 IC50 = 1250 nM T59328 C5EO6F 5328053 IC50 = 40 nM T59328 C3NP1J 5328054 IC50 = 65000 nM T59328 CFS1Q9 5328055 IC50 = 240 nM T59328 C5MB0W 5328056 IC50 = 90 nM T59328 C5U7TE 5328057 IC50 = 10000 nM T59328 CLG58H 5328058 IC50 = 15 nM T59328 CK3W0S 5328059 IC50 = 4700 nM T59328 CECV59 5328060 IC50 = 3710 nM T59328 C6QT8H 5328061 IC50 = 130 nM T59328 CL2KB9 5328062 IC50 = 670 nM T59328 CT87KZ 5328063 IC50 = 5250 nM T59328 CFSQ97 5328064 IC50 = 1550 nM T59328 CIWL47 5328065 IC50 = 5900 nM T59328 C4AY9I 5328066 IC50 = 69000 nM T59328 CN7I4H 5328067 IC50 = 1790 nM T59328 CA02CD 5328068 IC50 = 4860 nM T59328 C6MZ2K 5328069 IC50 = 840 nM T59328 C4CGO6 5328070 IC50 = 120 nM T59328 C68BQO 5328071 IC50 = 260 nM T59328 CEJB59 5328072 IC50 = 70 nM T59328 C1B7ZI 5328073 IC50 = 40 nM T59328 C0VL9E 5328074 IC50 > 10000 nM T59328 CW73VX 5328075 IC50 > 10000 nM T59328 CJ6CB8 5328076 IC50 > 10000 nM T59328 CJ6PO5 5328078 IC50 = 4250 nM T59328 C1N8WQ 5328079 IC50 = 10100 nM T59328 C58USW 5328080 IC50 > 10000 nM T59328 C5I8CA 5328081 IC50 = 1670 nM T59328 CM5EX7 5328082 IC50 = 1000 nM T59328 C1U0NE 5328083 IC50 = 2460 nM T59328 CRA1U0 5328084 IC50 = 10000 nM T59328 C1BC5V 5328085 IC50 = 1950 nM T59328 C5NKF7 5328086 IC50 = 8000 nM T59328 C6ID3P 5328087 IC50 = 100000 nM T59328 C6XJ8Q 5328088 IC50 = 2870 nM T59328 C7SC8N 5328089 IC50 > 100000 nM T59328 C94MXF 5328090 IC50 = 230 nM T59328 C8FI2S 5328091 IC50 > 10000 nM T59328 C0M5QH 5328092 IC50 > 10000 nM T59328 C05WQF 5328093 IC50 > 100000 nM T59328 CEB5H2 5328094 IC50 = 10000 nM T59328 C0XFQ1 5328095 IC50 > 100000 nM T59328 CCZ96X 5328096 IC50 = 1800 nM T59328 CW4XA5 5328097 IC50 = 3300 nM T59328 CHS5A1 5328098 IC50 > 100000 nM T59328 C4IJ7Z 5328099 IC50 = 3500 nM T59328 C4G6XV 5328100 Ki = 3100 nM T59328 CMTP83 5328101 IC50 = 4700 nM T59328 CH4P3L 5328102 IC50 = 13000 nM T59328 C5R9ZI 5328103 IC50 = 4600 nM T59328 CM06LQ 5328104 IC50 = 6900 nM T59328 CPT61U 5328112 IC50 = 450 nM T59328 CXR9K1 5328115 IC50 = 6200 nM T59328 CM0H5O 5328117 IC50 = 610 nM T59328 CDM98R 5328125 IC50 = 6680 nM T59328 CDY2O3 5328134 IC50 = 1300 nM T59328 CC1O0M 5328135 IC50 = 240 nM T59328 C14LVT 5328137 IC50 = 1000 nM T59328 COT45A 5328149 IC50 = 150 nM T59328 CF3AM9 5328157 IC50 = 980 nM T59328 CT9SO8 5328158 IC50 = 880 nM T59328 CJA36I 5328171 IC50 = 720 nM T59328 C5CZF2 5328186 IC50 = 55 nM T59328 CVF39K 5328187 IC50 = 770 nM T59328 C8SQG9 5328188 IC50 = 575.44 nM T59328 C2L4GQ 5328189 IC50 = 5000 nM T59328 C5L7OH 5328190 IC50 = 120 nM T59328 C6G8MS 5328191 IC50 = 100 nM T59328 CR6UC1 5328192 IC50 = 2 nM T59328 CSE29Z 5328193 IC50 = 0.25 nM T59328 CE2X5M 5328194 IC50 = 0.35 nM T59328 CDN5A9 5328195 IC50 = 3.3 nM T59328 CE3OP6 5328196 IC50 = 12000 nM T59328 CAU43H 5328197 IC50 = 6100 nM T59328 CR5Q3J 5328198 IC50 = 810 nM T59328 C9B8MI 5328199 IC50 = 540 nM T59328 C0V3QG 5328200 IC50 > 10000 nM T59328 C48GSA 5328201 IC50 = 0.89 nM T59328 C2TVO1 5328202 IC50 = 0.24 nM T59328 CQ3SK4 5328203 IC50 = 4 nM T59328 C3DXQ1 5328204 IC50 = 84 nM T59328 CL3X6O 5328205 IC50 = 12.02 nM T59328 CMQ0D5 5328207 IC50 = 40 nM T59328 C8VF0X 5328208 IC50 = 4 nM T59328 CASZ78 5328209 IC50 = 12 nM T59328 CCQX42 5328210 IC50 = 11 nM T59328 CEK4W5 5328211 IC50 = 162.18 nM T59328 CH89ZL 5328212 IC50 = 3.802 nM T59328 CB35RO 5328213 IC50 = 6.5 nM T59328 CX7CS9 5328214 IC50 = 53 nM T59328 CXWA71 5328215 IC50 = 68 nM T59328 CX4FR7 5328216 IC50 = 2000 nM T59328 CA6M1B 5328217 IC50 = 28 nM T59328 C1SR4I 5328218 IC50 = 15 nM T59328 CQ3MT4 5328219 IC50 = 25.12 nM T59328 C5W4EO 5328220 IC50 = 15 nM T59328 CPBJ63 5328221 IC50 = 0.1738 nM T59328 CA0E1F 5328222 IC50 = 105 nM T59328 CE9H1T 5328223 IC50 = 1370 nM T59328 CA4C8N 5328224 IC50 > 10000 nM T59328 CIEL17 5328225 IC50 > 10000 nM T59328 CCX4R2 5328226 IC50 = 463 nM T59328 CKY7Z5 5328227 IC50 = 152 nM T59328 CO12GB 5328228 IC50 = 0.67 nM T59328 CTV8F0 5328229 IC50 > 10000 nM T59328 CZG75R 5328230 IC50 = 128 nM T59328 COH17Q 5328231 IC50 = 0.072 nM T59328 CYU3Z1 5328232 IC50 = 113 nM T59328 CD8JS2 5328233 IC50 = 0.29 nM T59328 C5FY4G 5328234 IC50 = 0.01 nM T59328 C5GCU1 5328235 IC50 = 1.32 nM T59328 CJN72V 5328236 IC50 = 22 nM T59328 CV7UC8 5328237 IC50 = 203 nM T59328 CZE57H 5328238 IC50 = 29 nM T59328 C3TNY6 5328239 IC50 = 272 nM T59328 C5LS7N 5328240 IC50 = 44 nM T59328 C4S0YJ 5328241 IC50 = 0.34 nM T59328 CP4Y5S 5328242 IC50 = 0.44 nM T59328 C3EF7M 5328243 IC50 = 0.39 nM T59328 CAE24W 5328246 IC50 = 1.7 nM T59328 CH62XU 5328247 IC50 = 1460 nM T59328 C7XLU4 5328248 IC50 = 100 nM T59328 CS60WL 5328249 IC50 = 35.48 nM T59328 C6CU9X 5328250 IC50 = 29 nM T59328 CRW56D 5328251 IC50 = 13 nM T59328 CHZ78I 5328252 IC50 = 16 nM T59328 C1LX5E 5328253 IC50 = 14 nM T59328 C3EB6U 5328254 IC50 = 39 nM T59328 CUAH85 5328256 IC50 = 2030 nM T59328 CWCJ02 5328257 IC50 = 51 nM T59328 CC0F5Z 5328258 IC50 = 0.13 nM T59328 CY0AH6 5328259 IC50 = 40 nM T59328 C8UG0Z 5328260 IC50 = 124 nM T59328 CVK13Z 5328261 IC50 = 0.006 nM T59328 CVT30D 5328262 IC50 = 2.63 nM T59328 C4ML9Z 5328263 IC50 = 2.3 nM T59328 CZU8N4 5328264 IC50 = 9 nM T59328 CJU52L 5328265 IC50 > 10 nM T59328 C7QH8D 5328266 IC50 = 688 nM T59328 C5C4BE 5328267 IC50 = 954.99 nM T59328 CCN5Y6 5328268 IC50 = 684 nM T59328 CE1Q2B 5328269 IC50 = 52 nM T59328 CA4R3X 5328270 IC50 = 331.13 nM T59328 C8BP2W 5328271 IC50 = 263 nM T59328 C5YRH9 5328272 IC50 = 603 nM T59328 C5O7VR 5328273 IC50 = 34 nM T59328 CE3JU1 5328274 IC50 = 53 nM T59328 C7WD6E 5328275 IC50 = 18 nM T59328 C1ORZ0 5328276 IC50 = 44 nM T59328 C2L3RB 5328277 IC50 = 3.1 nM T59328 CD20TF 5328278 IC50 = 9.6 nM T59328 CQO15H 5328279 IC50 = 4.3 nM T59328 CNEF93 5328280 IC50 = 0.37 nM T59328 CR2W7Q 5328281 IC50 = 12 nM T59328 CA2CP7 5328282 IC50 = 39.81 nM T59328 CS16CZ 5328283 IC50 = 3.7 nM T59328 CEF8A6 5328284 IC50 = 52.48 nM T59328 CUFW39 5328285 IC50 = 21.88 nM T59328 C1PC0U 5328286 IC50 = 1.6 nM T59328 CI7H3A 5328287 IC50 = 41 nM T59328 C8O2FY 5328288 IC50 = 21 nM T59328 CQ1OD4 5328289 IC50 = 3.7 nM T59328 C0W1HD 5328290 IC50 = 77.62 nM T59328 C0R1WK 5328291 IC50 = 5.1 nM T59328 C0QUZ5 5328292 IC50 = 135 nM T59328 CTI8W5 5328293 IC50 = 9.7 nM T59328 C8THM7 5328294 IC50 = 4.8 nM T59328 CJY1D0 5328295 IC50 = 81 nM T59328 C7FQ0J 5328296 IC50 = 3.388 nM T59328 CI32AD 5328297 IC50 = 0.72 nM T59328 C49IVK 5328298 IC50 = 0.24 nM T59328 C03MPD 5328299 IC50 = 2.57 nM T59328 CN7T3V 5328300 IC50 = 0.92 nM T59328 CL6HI8 5328301 IC50 = 3.2 nM T59328 C0JO8H 5328302 IC50 = 14 nM T59328 CVZQ92 5328303 IC50 = 12 nM T59328 CMV6R1 5328304 IC50 = 4.786 nM T59328 CSGC46 5328305 IC50 = 3.2 nM T59328 C0HIY2 5328306 IC50 = 44.67 nM T59328 C75QGA 5328307 IC50 = 8.71 nM T59328 CED9Z1 5328308 IC50 = 7.4 nM T59328 C5LC3J 5328309 IC50 = 8.318 nM T59328 C2RB9W 5328310 IC50 = 39.81 nM T59328 CT1V0S 5328311 IC50 = 3.236 nM T59328 CH1RI6 5328312 IC50 = 1.9 nM T59328 C82PRW 5328313 IC50 = 5.4 nM T59328 C5IN3X 5328314 IC50 = 0.74 nM T59328 CZ1VX5 5328315 IC50 = 4.898 nM T59328 CE6H9B 5328316 IC50 = 9.12 nM T59328 CH1ZV3 5328317 IC50 = 1.2 nM T59328 CEX9D0 5328318 IC50 = 7.1 nM T59328 CW4MH8 5328319 IC50 = 0.51 nM T59328 C2X4IR 5328320 IC50 = 0.91 nM T59328 C8CT3Z 5328321 IC50 = 1.5 nM T59328 C1UC9A 5328322 IC50 = 0.61 nM T59328 C4MO0D 5328323 IC50 = 0.2818 nM T59328 CLGB27 5328324 IC50 = 15.85 nM T59328 CY0AM6 5328325 IC50 = 1.4 nM T59328 CX7JZ8 5328326 IC50 = 1.413 nM T59328 C4CJW1 5328327 IC50 = 5.37 nM T59328 C80JRW 5328328 IC50 = 9.3 nM T59328 CWM81T 5328329 IC50 = 5.6 nM T59328 CZ8GQ5 5328330 IC50 = 3.5 nM T59328 C27YZX 5328331 IC50 = 7.2 nM T59328 C4BXI1 5328332 IC50 = 2550 nM T59328 CF8X6A 5328333 IC50 = 13 nM T59328 CHR91V 5328334 IC50 = 83.18 nM T59328 CZ1M2D 5328335 IC50 = 1.5 nM T59328 CSH09Q 5328336 IC50 = 0.76 nM T59328 C5S9YM 5328337 IC50 = 0.95 nM T59328 CFR57D 5328338 IC50 = 3.8 nM T59328 CUN2R4 5328339 IC50 = 35 nM T59328 C0NY7V 5328340 IC50 = 0.81 nM T59328 C0LDH1 5328341 IC50 = 2.9 nM T59328 CQ6ZM5 5328342 IC50 = 0.2512 nM T59328 CC2VT4 5328343 IC50 = 2.3 nM T59328 CUY75Z 5328344 IC50 = 380 nM T59328 CA6KZ4 5328345 IC50 = 17 nM T59328 CB3OP9 5328346 IC50 = 4.3 nM T59328 C1R7LX 5328347 IC50 = 4 nM T59328 CA1VR6 5328348 IC50 = 2.3 nM T59328 CK92CS 5328349 IC50 = 3 nM T59328 COI17R 5328350 IC50 = 0.19 nM T59328 C34OXD 5328351 IC50 = 0.22 nM T59328 CB4AJ3 5328352 IC50 = 0.18 nM T59328 C7ABZ1 5328353 IC50 = 0.56 nM T59328 CDV19S 5328354 IC50 = 1.1 nM T59328 CN62LQ 5328355 IC50 = 1.2 nM T59328 CIW27V 5328356 IC50 = 1.8 nM T59328 C1D0YT 5328357 IC50 = 4.6 nM T59328 C0X4VK 5328358 IC50 = 1.7 nM T59328 CV1L9N 5328359 IC50 = 8.1 nM T59328 CC4O6Y 5328360 IC50 = 0.65 nM T59328 CE3UW4 5328361 IC50 = 1 nM T59328 CU65HL 5328363 IC50 = 0.93 nM T59328 C7L1MN 5328364 IC50 = 230 nM T59328 C6S4LT 5328365 IC50 = 1.5 nM T59328 CG4RZ8 5328366 IC50 = 1.2 nM T59328 C6K4VL 5328367 IC50 = 0.78 nM T59328 CYLS53 5328368 IC50 = 1.7 nM T59328 CJY62E 5328369 IC50 = 102 nM T59328 C5EO4G 5328370 IC50 = 0.28 nM T59328 CP37XG 5328371 IC50 = 0.44 nM T59328 C0X8JK 5328372 IC50 = 449 nM T59328 C0EFY7 5328373 IC50 = 0.19 nM T59328 C7R3YC 5328374 IC50 = 1.1 nM T59328 C8IXG0 5328375 IC50 = 3.1 nM T59328 CE4R1Q 5328376 IC50 = 0.45 nM T59328 C0ON1H 5328377 IC50 = 2.8 nM T59328 CWPM74 5328378 IC50 = 1.5 nM T59328 C2QNS7 5328379 IC50 = 1.8 nM T59328 C3MHX9 5328380 IC50 = 1.3 nM T59328 CG0W7E 5328381 IC50 = 117 nM T59328 CJF0H4 5328382 IC50 = 1 nM T59328 CM96IG 5328383 IC50 = 11 nM T59328 C2REG3 5328387 IC50 = 419 nM T59328 CTBV20 5328388 IC50 = 50 nM T59328 CG3J4S 5328389 IC50 > 100000 nM T59328 CJY35F 5328391 IC50 = 264 nM T59328 C5FY3T 5328392 IC50 = 31 nM T59328 CXNL13 5328393 IC50 = 742 nM T59328 CF7J4M 5328394 IC50 = 4100 nM T59328 CF5SL0 5328396 IC50 = 147 nM T59328 CDEY49 5328397 IC50 = 1.2 nM T59328 C51IFH 5328398 IC50 = 4270 nM T59328 CEG9H2 5328399 IC50 = 191 nM T59328 C84GLZ 5328400 IC50 = 538 nM T59328 C6JA7G 5328401 IC50 = 1.8 nM T59328 CO17CE 5328407 IC50 = 2.1 nM T59328 CBO8C1 5328408 IC50 = 47 nM T59328 C61RXT 5328409 IC50 = 0.27 nM T59328 CVED61 5328412 IC50 = 42 nM T59328 CR6LU1 5328414 IC50 = 80 nM T59328 C1GL9F 5328416 IC50 = 19.8 nM T59328 CU2N1B 5328422 IC50 > 1000 nM T59328 CV2D5L 5328423 IC50 = 732 nM T59328 C46BDX 5328425 IC50 = 740 nM T59328 CJN93G 5328535 IC50 = 14900 nM T59328 CIV92Z 5328536 IC50 > 100000 nM T59328 CW8B1J 5328537 IC50 = 100000 nM T59328 CPN2E4 5328538 IC50 > 100000 nM T59328 CLQ9B1 5328539 IC50 = 1620 nM T59328 CA7LK0 5328540 IC50 = 6700 nM T59328 CW59PN 5328541 IC50 > 100000 nM T59328 CWB7K0 5328542 IC50 > 100000 nM T59328 C3UWT2 5328543 IC50 = 6700 nM T59328 C5FA3P 5328544 IC50 > 100000 nM T59328 C9DL4S 5328545 IC50 > 100000 nM T59328 C2PF4N 5328546 IC50 > 100000 nM T59328 C6UWZ8 5328547 IC50 > 100000 nM T59328 C9LMP7 5328548 IC50 > 100000 nM T59328 C3D5KN 5328549 IC50 > 100000 nM T59328 CL7JE8 5328550 IC50 = 10200 nM T59328 CV08ZJ 5328551 IC50 = 53000 nM T59328 CEQ5A8 5328552 IC50 = 14000 nM T59328 C0MP1C 5328553 IC50 = 18000 nM T59328 C3QA9X 5328554 IC50 = 33000 nM T59328 C6DN3V 5328555 IC50 > 100000 nM T59328 C6CMP2 5328556 IC50 = 9300 nM T59328 CQA3V1 5328557 IC50 = 35000 nM T59328 C3UAX9 5328558 IC50 = 4200 nM T59328 CS8A1P 5328559 IC50 = 3100 nM T59328 C3NC0W 5328560 IC50 = 21000 nM T59328 CXOP18 5328561 IC50 > 100000 nM T59328 C09UBN 5328562 IC50 = 8400 nM T59328 C71VUG 5328563 IC50 = 2900 nM T59328 COGL89 5328564 IC50 = 1500 nM T59328 CP5YX1 5328565 IC50 = 18000 nM T59328 C3WH4C 5328566 IC50 = 8300 nM T59328 C0QYJ7 5328567 IC50 > 100000 nM T59328 CHW4Q7 5328568 IC50 > 100000 nM T59328 CB9UI5 5328569 IC50 = 38000 nM T59328 CVEY01 5328570 IC50 = 32000 nM T59328 C3U1QJ 5328571 IC50 = 47000 nM T59328 CP5H9N 5328572 IC50 = 89000 nM T59328 C64XYH 5328573 IC50 = 16000 nM T59328 CBE9M4 5328574 IC50 = 9400 nM T59328 C5QE9H 5328575 IC50 = 68000 nM T59328 CE9PW4 5328576 IC50 = 12000 nM T59328 CJ78UZ 5328577 IC50 = 25000 nM T59328 C9S1MH 5328578 IC50 = 850 nM T59328 CE62YD 5328579 IC50 = 44000 nM T59328 C72KTF 5328580 IC50 = 7400 nM T59328 CG38AH 5328581 IC50 = 100000 nM T59328 C5HB9Z 5328582 IC50 = 8500 nM T59328 CGDE60 5328583 IC50 = 24000 nM T59328 COF98M 5328584 IC50 = 51000 nM T59328 C23LDB 5328585 IC50 > 100000 nM T59328 CXN72C 5328586 IC50 = 28000 nM T59328 CAT93L 5328587 IC50 = 14000 nM T59328 CA9PL4 5328588 IC50 = 100000 nM T59328 CQDX90 5328589 IC50 = 100000 nM T59328 CLZ2T7 5328590 IC50 = 22000 nM T59328 CMP24I 5328591 IC50 = 100000 nM T59328 C0TX2I 5328592 IC50 = 10000 nM T59328 C9JLN6 5328593 IC50 = 100000 nM T59328 C42LEK 5328594 IC50 > 100000 nM T59328 CVF12E 5328595 IC50 > 100000 nM T59328 CGN3C9 5328596 IC50 = 20000 nM T59328 C91NOL 5328597 IC50 > 100000 nM T59328 C0PB9W 5328598 IC50 = 4300 nM T59328 C9P3LY 5328599 IC50 = 11400 nM T59328 CQNB13 5328600 IC50 > 100000 nM T59328 CK7IA1 5328601 IC50 > 100000 nM T59328 CNI91T 5328602 IC50 = 5300 nM T59328 C3AW9S 5328603 IC50 = 40500 nM T59328 CWEA08 5328604 IC50 > 100000 nM T59328 CCM96I 5328605 IC50 = 54100 nM T59328 C9NVC5 5328606 IC50 = 5000 nM T59328 CDX4Z7 5328607 IC50 > 100000 nM T59328 CB1S3D 5328608 IC50 > 100000 nM T59328 C7WL3M 5328609 IC50 = 3600 nM T59328 C69QIE 5328610 IC50 > 100000 nM T59328 C09SPY 5328611 IC50 = 44000 nM T59328 CO2CR8 5328612 IC50 > 100000 nM T59328 CR3W8H 5328613 IC50 > 100000 nM T59328 CB2HD4 5328614 IC50 = 6500 nM T59328 C5GWD8 5328615 IC50 = 9900 nM T59328 C0MU7G 5328616 IC50 = 100000 nM T59328 CH1X6G 5328617 IC50 = 22300 nM T59328 CR02JQ 5328618 IC50 = 1000 nM T59328 CP8G4Z 5328619 IC50 > 100000 nM T59328 C8YS2H 5328620 IC50 > 100000 nM T59328 CM80FN 5328621 IC50 > 100000 nM T59328 C16JYR 5328622 IC50 > 100000 nM T59328 CL6QD5 5328623 IC50 > 100000 nM T59328 CFB26C 5328624 IC50 > 100000 nM T59328 C38PSR 5328744 IC50 > 250000 nM T59328 CJLU79 5328746 IC50 = 532000 nM T59328 CGM84A 5328747 IC50 = 800000 nM T59328 C71JTL 5328748 IC50 = 820000 nM T59328 CA9RY2 5328749 IC50 = 1480000 nM T59328 C2HDP0 5328750 IC50 = 1800000 nM T59328 C7LS0I 5328751 IC50 = 2200000 nM T59328 C6J4FI 5328752 IC50 > 2500000 nM T59328 CY9UG7 5328754 IC50 = 2500 nM T59328 CY8U9E 5328756 IC50 = 12500 nM T59328 CSZK53 5328757 IC50 = 26000 nM T59328 C46ZGF 5328758 IC50 = 60000 nM T59328 CX2G6U 5328759 IC50 = 1200000 nM T59328 CND59O 5328761 IC50 = 560 nM T59328 C68MGU 5328762 IC50 = 880 nM T59328 CN8L0R 5328764 IC50 = 1540 nM T59328 C2B0HF 5328765 IC50 = 2000 nM T59328 C4HNQ7 5328766 IC50 = 3100 nM T59328 CLQ73F 5328767 IC50 = 19054.61 nM T59328 C3F7YW 5328770 IC50 = 700 nM T59328 C67KXB 5328771 IC50 = 700 nM T59328 CJ6U2C 5328773 IC50 < 625 nM T59328 C7VW9X 5328774 IC50 = 2089.3 nM T59328 CSL05I 5328775 IC50 = 3000 nM T59328 C5ZV9K 5328776 IC50 = 1530 nM T59328 C3GRB0 5328777 IC50 = 1700 nM T59328 CI97TH 5328778 IC50 = 1700 nM T59328 CMX61C 5328780 IC50 = 4300 nM T59328 CED31Y 5328781 IC50 = 5100 nM T59328 CZ9Y4I 5328782 Ki = 240000 nM T59328 CBNU15 5328783 Ki = 150000 nM T59328 C2E4VB 5328784 Ki = 143000 nM T59328 CB2W9A 5328785 Ki = 49000 nM T59328 C75XMH 5328786 Ki = 24000 nM T59328 CH86SJ 5328787 Ki = 20000 nM T59328 CD8SN1 5328788 Ki = 10000 nM T59328 CJC2Z1 5328789 IC50 = 1300000 nM T59328 CF3MR6 5328790 IC50 = 264000 nM T59328 C94SUH 5328791 IC50 = 165000 nM T59328 C9PCS3 5328792 IC50 = 47000 nM T59328 C4N0CE 5328793 IC50 = 30000 nM T59328 CS98WX 5328794 IC50 > 1250000 nM T59328 CEA86M 5328795 Ki = 341000 nM T59328 CNB7Q3 5328796 IC50 = 800000 nM T59328 CGY6U3 5328797 Ki = 360000 nM T59328 CP50YI 5328798 IC50 = 500000 nM T59328 CD6JM3 5328799 IC50 = 450000 nM T59328 C5HQJ7 5328800 IC50 = 230000 nM T59328 CS09OR 5328801 Ki = 4500 nM T59328 CD6SC0 5328802 IC50 = 50000 nM T59328 C46UBD 5328805 IC50 = 60000 nM T59328 CR4K3Z 5328806 IC50 = 2500 nM T59328 CYO4C9 5328808 IC50 = 1000 nM T59328 CB8QZ6 5328809 IC50 = 500 nM T59328 C8M2UN 5328810 IC50 = 1360000 nM T59328 CLQA04 5328811 IC50 = 2400000 nM T59328 C5H3UK 5328812 Ki = 24000 nM T59328 CWJQ49 5328813 IC50 = 225000 nM T59328 C69RVL 5328814 IC50 = 350000 nM T59328 CU73YL 5328815 IC50 = 1400000 nM T59328 CEUV72 5328835 IC50 > 1000000 nM T59328 C2IN6M 5328838 IC50 = 416.87 nM T59328 CH6F9K 5328839 IC50 = 977.24 nM T59328 C7YRI8 5328840 IC50 = 90 nM T59328 CIQ54V 5328841 IC50 = 181.97 nM T59328 CCUR96 5328842 IC50 = 1445.44 nM T59328 CXH6C3 5328843 IC50 = 50118.72 nM T59328 CI9M3J 5328844 IC50 = 741.31 nM T59328 CB8RH3 5328845 IC50 = 14125.38 nM T59328 CJO6F4 5328846 IC50 = 47863.01 nM T59328 C2TQ4I 5328847 IC50 = 7413.1 nM T59328 C3QYM2 5328848 IC50 = 812.83 nM T59328 CU16VD 5328849 IC50 = 851.14 nM T59328 CX2CO0 5328850 IC50 = 870.96 nM T59328 CQK10C 5328851 IC50 = 5170 nM T59328 C0G6RT 5328852 IC50 = 13803.84 nM T59328 C9BYN7 5328853 IC50 = 6309.57 nM T59328 CZ3XY7 5328854 IC50 = 2754.23 nM T59328 C4K2ST 5328855 IC50 = 7762.47 nM T59328 CK6HN0 5328856 IC50 = 1778.28 nM T59328 CM60SD 5328857 IC50 = 9120.11 nM T59328 CL21YK 5328858 IC50 = 3162.28 nM T59328 CD1R8Q 5328859 IC50 = 16982.44 nM T59328 CY5MV7 5328860 IC50 = 758.58 nM T59328 C36EMZ 5328861 IC50 = 1479.11 nM T59328 CIXV80 5328863 IC50 = 229.09 nM T59328 CCE96Z 5328864 IC50 = 363.08 nM T59328 CMV0J2 5328865 IC50 = 61659.5 nM T59328 C47VGY 5328866 IC50 = 6606.93 nM T59328 CLOF23 5328867 IC50 = 4168.69 nM T59328 C3UBZ5 5328868 IC50 = 158.49 nM T59328 C5XM1A 5328869 IC50 = 831.76 nM T59328 C80RXA 5328870 IC50 = 616.6 nM T59328 C0KX1O 5328871 IC50 = 2187.76 nM T59328 CFIH48 5328872 IC50 = 69183.1 nM T59328 CBC41T 5328873 IC50 = 33113.11 nM T59328 CDG14R 5328874 IC50 = 21379.62 nM T59328 C5E0TK 5328877 IC50 = 3388.44 nM T59328 CC93DK 5328878 IC50 = 33884.42 nM T59328 C8F2JU 5328879 IC50 = 15135.61 nM T59328 C15RWZ 5328881 IC50 = 6760.83 nM T59328 CC3JI8 5328882 IC50 = 1096.48 nM T59328 CX18GK 5328883 IC50 = 6760.83 nM T59328 CYJ3W2 5328884 IC50 = 5128.61 nM T59328 CN5PO1 5328885 IC50 = 70794.58 nM T59328 C2PSJ1 5328886 IC50 = 89125.09 nM T59328 CT1QC6 5328954 IC50 = 6 nM T59328 C41BJK 5328955 IC50 = 12 nM T59328 CUW4V3 5328956 IC50 = 62 nM T59328 CI3Q6X 5328957 IC50 = 85 nM T59328 C0AF9T 5328958 IC50 = 97 nM T59328 C8A4XJ 5328959 IC50 = 71 nM T59328 CTN9X5 5328960 IC50 = 57 nM T59328 CP6G8R 5328961 IC50 = 20 nM T59328 CAQM41 5328962 IC50 = 95 nM T59328 CDJ8B5 5328964 IC50 = 65 nM T59328 C94KSU 5328965 IC50 = 9 nM T59328 C1W0DS 5328966 IC50 = 65 nM T59328 CX5S2M 5328967 IC50 = 59 nM T59328 CHL05B 5328968 IC50 = 2 nM T59328 CXN2Y0 5328969 IC50 = 0.22 nM T59328 C6BM9P 5328970 IC50 = 73 nM T59328 CR3GV8 5328971 IC50 = 90 nM T59328 CJU57A 5328972 IC50 = 106 nM T59328 CJ42FQ 5328973 IC50 = 74 nM T59328 CKA09Y 5328974 IC50 = 203 nM T59328 C92KTO 5328975 IC50 = 131 nM T59328 C4KI5U 5328976 IC50 = 85 nM T59328 CI36GZ 5328977 IC50 = 62 nM T59328 CU4W7S 5328978 IC50 = 14 nM T59328 C39VSH 5328979 IC50 = 68 nM T59328 C9U5YF 5328980 IC50 = 1124 nM T59328 CY4B5J 5328981 IC50 = 16 nM T59328 C03WIS 5328982 IC50 = 0.55 nM T59328 CG3KL4 5328983 IC50 = 1132 nM T59328 CV5KY4 5328984 IC50 = 115 nM T59328 CUJ6G5 5328985 IC50 = 107 nM T59328 CLP07T 5328986 IC50 = 250 nM T59328 CD60RC 5328987 IC50 = 215 nM T59328 CK15AU 5328988 IC50 = 269 nM T59328 C7R2EK 5328989 IC50 = 194 nM T59328 CFW19M 5329009 IC50 = 1 nM T59328 CZU0K3 5329011 IC50 = 100 nM T59328 C1XJL0 5329019 IC50 = 300 nM T59328 C9SZ4Q 5329020 IC50 = 100 nM T59328 C3VHF6 5329026 IC50 = 300 nM T59328 C9VX8C 5329040 IC50 = 1400 nM T59328 CK6T4U 5329042 IC50 = 400 nM T59328 CA81XO 5329045 IC50 = 450 nM T59328 C4T3MO 5329046 IC50 = 300 nM T59328 CQ15KR 5329049 IC50 = 450 nM T59328 C49KNS 5329050 IC50 = 500 nM T59328 C3C1EZ 5329051 IC50 = 400 nM T59328 C0H5XL 5329052 IC50 = 300 nM T59328 CW0KA8 5329053 IC50 = 200 nM T59328 COEN93 5329054 IC50 = 80 nM T59328 CATX52 5329055 IC50 = 100 nM T59328 CEQP41 5329056 IC50 = 150 nM T59328 CDV4C9 5329057 IC50 = 100 nM T59328 CH26SN 5329069 IC50 = 0.91 nM T59328 C7RF9L 5329070 IC50 = 0.17 nM T59328 CGTA78 5329071 IC50 = 1.6 nM T59328 CBV46K 5329072 IC50 = 0.5 nM T59328 CXG29Q 5329074 IC50 = 1.75 nM T59328 C6MX8O 5329075 IC50 = 27 nM T59328 CN02JA 5329077 IC50 = 9.1 nM T59328 CF0U7Z 5329078 IC50 = 1039 nM T59328 CE0UT9 5329079 IC50 = 0.37 nM T59328 CJFE40 5329080 IC50 = 2.7 nM T59328 CS84JW 5329081 IC50 = 1.5 nM T59328 C71GUX 5329082 IC50 = 4.2 nM T59328 C07AVK 5329083 IC50 = 2.7 nM T59328 CHS1I6 5329084 IC50 = 3.3 nM T59328 C5JL2Y 5329085 IC50 = 2.4 nM T59328 CT4U5F 5329086 IC50 = 0.44 nM T59328 CBY4R5 5329087 IC50 = 1.1 nM T59328 C53HOJ 5329088 IC50 = 0.73 nM T59328 C2P3EO 5329089 IC50 = 0.81 nM T59328 C61NGH 5329090 IC50 = 14 nM T59328 CUZ82W 5329091 IC50 = 1.45 nM T59328 CAV71E 5329092 IC50 = 0.6026 nM T59328 C0OD8J 5329093 IC50 = 0.76 nM T59328 C0A8HY 5329094 IC50 = 2.7 nM T59328 CPH8Q3 5329095 IC50 = 93.5 nM T59328 CG2QX5 5329096 IC50 = 0.4266 nM T59328 CE48UM 5329097 IC50 = 340 nM T59328 C9I7WT 5329100 IC50 > 20000 nM T59328 CMWB28 5329101 IC50 > 20000 nM T59328 CGX50J 5329104 IC50 = 10000 nM T59328 C2VX0H 5329105 IC50 > 20000 nM T59328 CK71MQ 5329106 IC50 > 20000 nM T59328 C6YRH8 5329108 IC50 > 20000 nM T59328 CFP59Y 5329109 IC50 > 20000 nM T59328 CSY10K 5329111 IC50 = 5530 nM T59328 C0JW3Y 5329134 IC50 = 28800 nM T59328 CO7J2A 5329135 IC50 > 50000 nM T59328 CQ4TP5 5329136 IC50 = 49200 nM T59328 CXQC42 5329137 IC50 > 50000 nM T59328 CT94JS 5329138 IC50 > 50000 nM T59328 CNH06M 5329139 IC50 > 100000 nM T59328 CRY4Z2 5329140 IC50 > 50000 nM T59328 CAPE50 5329141 IC50 > 50000 nM T59328 CFU58A 5329142 IC50 = 21800 nM T59328 C5Q8XK 5329143 IC50 = 30500 nM T59328 C8PX4D 5329144 IC50 = 19200 nM T59328 C6USQ5 5329145 IC50 = 22800 nM T59328 C56LWT 5329146 IC50 > 100000 nM T59328 CZ16MN 5329147 IC50 > 50000 nM T59328 CAN16I 5329148 IC50 > 50000 nM T59328 CG4NC2 5329149 IC50 > 100000 nM T59328 CIW70H 5329150 IC50 = 21900 nM T59328 C5FT6A 5329151 IC50 = 24100 nM T59328 CB0N4L 5329152 IC50 = 31300 nM T59328 COFP24 5329153 IC50 > 50000 nM T59328 CGWD98 5329154 IC50 > 100000 nM T59328 C4PD0K 5329156 IC50 > 100000 nM T59328 C0RWT8 5329157 IC50 > 100000 nM T59328 C3MU5S 5329158 IC50 > 100000 nM T59328 CN6O4R 5329159 IC50 > 100000 nM T59328 CG68DI 5329160 IC50 > 100000 nM T59328 CYR7V0 5329161 IC50 > 100000 nM T59328 C9BXE2 5329162 IC50 > 100000 nM T59328 CY4V5Z 5329163 IC50 > 100000 nM T59328 CI64YA 5329164 IC50 > 100000 nM T59328 C2ZV0O 5329165 IC50 = 29100 nM T59328 CAB53L 5329166 IC50 = 56500 nM T59328 CTW9R8 5329167 IC50 > 100000 nM T59328 C8A3TJ 5329168 IC50 > 100000 nM T59328 CVTD82 5329169 IC50 = 8880 nM T59328 CQ5WK1 5329170 IC50 > 100000 nM T59328 CNC9T7 5329171 IC50 > 100000 nM T59328 C6L0UW 5329229 IC50 > 20000 nM T59328 C1DBV6 5329230 IC50 = 180 nM T59328 CLKM80 5329231 IC50 = 200 nM T59328 CTQ18A 5329232 IC50 = 7820 nM T59328 CM5KG6 5329233 IC50 = 4.7 nM T59328 CQG6R2 5329234 IC50 = 29 nM T59328 CJ3A9I 5329235 IC50 = 22 nM T59328 CPS7X1 5329236 IC50 = 6.5 nM T59328 CAN60T 5329237 IC50 > 20000 nM T59328 CY15JP 5329238 IC50 = 5310 nM T59328 C41UBI 5329239 IC50 = 40 nM T59328 C6VQ9F 5329240 IC50 = 2.8 nM T59328 C8WS5K 5329241 IC50 = 210 nM T59328 CI26UN 5329242 IC50 = 410 nM T59328 C6PJ2R 5329243 IC50 = 13 nM T59328 C0OKB7 5329244 IC50 = 200 nM T59328 C78ZNL 5329245 IC50 = 5.9 nM T59328 CWL5S4 5329246 IC50 = 0.45 nM T59328 C4X3OE 5329248 IC50 = 450 nM T59328 CK8FH6 5329249 IC50 = 1410 nM T59328 CN5B6C 5329250 IC50 = 100 nM T59328 CQ0B6E 5329251 IC50 = 100 nM T59328 C4KO3N 5329252 IC50 = 200 nM T59328 C6MZF8 5329253 IC50 > 20000 nM T59328 CO1U8I 5329254 IC50 = 340 nM T59328 C54NXZ 5329255 IC50 = 400 nM T59328 CN4MD2 5329256 IC50 = 10000 nM T59328 CJ9O8L 5329257 IC50 = 4300 nM T59328 C0WJ6Y 5329258 IC50 = 5000 nM T59328 CA6H2Y 5329259 IC50 = 700 nM T59328 CFP2O6 5329260 IC50 = 700 nM T59328 CV6KI2 5329261 IC50 = 1300 nM T59328 CLK4V3 5329262 IC50 = 6000 nM T59328 CXUV69 5329263 IC50 = 12500 nM T59328 CSV71T 5329264 IC50 = 19000 nM T59328 C9S6OV 5329266 IC50 = 2200 nM T59328 CIV10W 5329267 IC50 = 2200 nM T59328 C96PSZ 5329268 IC50 = 4000 nM T59328 CJR4T0 5329269 IC50 > 100000 nM T59328 CP20TG 5329270 IC50 = 2000 nM T59328 C8R2YT 5329271 IC50 = 1400 nM T59328 C2AR4T 5329272 IC50 = 940 nM T59328 CD6NV0 5329475 IC50 = 34.67 nM T59328 CA78HB 5329476 IC50 = 81.28 nM T59328 C0OAR2 5329477 IC50 = 70.79 nM T59328 C8A3GZ 5329478 IC50 = 537.03 nM T59328 C78XVZ 5329479 IC50 = 7.943 nM T59328 CQ39FM 5329480 IC50 = 10 nM T59328 CVS3Z1 5329481 IC50 = 97.72 nM T59328 CW2UJ7 5329482 IC50 = 263 nM T59328 CY14AK 5329483 IC50 = 74 nM T59328 CIT24W 5329484 IC50 = 68 nM T59328 CDZ6R5 5329485 IC50 = 79 nM T59328 C3LSH8 5329486 IC50 = 104 nM T59328 CGZA12 5329487 IC50 = 830 nM T59328 CV9L1J 5329488 IC50 = 74.13 nM T59328 CJD92I 5329489 IC50 = 11 nM T59328 CS1HF6 5329490 IC50 = 19.95 nM T59328 CX4L0Q 5329491 IC50 = 93 nM T59328 C9C3SD 5329492 IC50 = 27 nM T59328 CDRM58 5329493 IC50 = 24 nM T59328 CS2HM9 5329714 IC50 > 50000 nM T59328 CM9V8E 5329715 IC50 > 50000 nM T59328 CB0QZ2 5330117 IC50 > 1000 nM T59328 C7QZL3 5330118 IC50 > 1000 nM T59328 CNR9B8 5330119 IC50 > 1000 nM T59328 CXY2I9 5330120 IC50 > 1000 nM T59328 CDF96J 5330121 IC50 > 1000 nM T59328 C7BPR2 5330122 IC50 > 1000 nM T59328 CC4ZJ3 5330123 IC50 > 1000 nM T59328 CLV0T6 5330124 IC50 > 1000 nM T59328 CZ3LK2 5330387 IC50 = 1360 nM T59328 CRU94N 5330388 IC50 = 7400 nM T59328 CDB68F 5330389 IC50 > 10000 nM T59328 C7CX0H 5330390 IC50 > 10000 nM T59328 C5SY4O 5330420 IC50 = 2000 nM T59328 CUEZ35 5330437 IC50 = 2700 nM T59328 C94GRU 5330453 IC50 = 3000 nM T59328 CC2E4Q 5330468 IC50 = 7100 nM T59328 C1YWE0 5330475 IC50 = 27000 nM T59328 C9NBG7 5330546 IC50 > 10000 nM T59328 CF01JS 5330804 IC50 = 8400 nM T59328 C3U0TG 5330830 IC50 > 100000 nM T59328 CL1FH5 5330832 IC50 > 100000 nM T59328 C1P2ZA 5330847 IC50 > 100000 nM T59328 CM47KI 5351344 IC50 > 10000 nM T59328 CYXI29 5353388 IC50 = 400 nM T59328 CJ5A1W 5353391 IC50 = 100 nM T59328 CHD1L6 5353609 IC50 = 20 ug.mL-1 T59328 CQ12UT 5353911 IC50 = 0.1 ug.mL-1 T59328 CDQ3M7 5359485 IC50 = 5.5 ug.mL-1 T59328 C54BYP 5360741 IC50 = 1.7 ug.mL-1 T59328 C6REP3 5371842 IC50 = 38460 nM T59328 CB8DX4 5371857 IC50 = 29850 nM T59328 C23XEH 5386499 IC50 > 100 ug.mL-1 T59328 CL5W9P 5386517 IC50 > 10 ug.mL-1 T59328 C63YGX 5386800 IC50 = 0.3 ug.mL-1 T59328 C0SO6F 5388678 IC50 = 10000 nM T59328 C6RAT9 5388682 IC50 = 7000 nM T59328 C2O9ZG 5391486 IC50 = 31800 nM T59328 CD65JT 5427216 IC50 > 100000 nM T59328 CPB95V 5427224 IC50 > 100000 nM T59328 CL27VO 5467485 IC50 = 20300 nM T59328 CRKI23 5468831 IC50 = 5800 nM T59328 CZ0NU2 5481591 IC50 > 1000 nM T59328 CCT39K 5703472 IC50 = 10100 nM T59328 CA6L5V 5707304 IC50 > 100000 nM T59328 C43YGE 5713379 IC50 > 100000 nM T59328 CS24NJ 5775636 IC50 = 9000 nM T59328 CT8U7I 5874584 IC50 > 100000 nM T59328 CO6KI2 5930298 IC50 > 10000 nM T59328 CRW23P 5941457 IC50 = 400 nM T59328 CM8LW9 6036100 IC50 > 100000 nM T59328 CPU89Q 6082393 IC50 = 35000 nM T59328 C7MD9J 6091659 IC50 = 18600 nM T59328 C3R9VW 6105823 IC50 = 3 ug.mL-1 T59328 C9XV5P 6398579 IC50 = 1300000 nM T59328 C0IYS8 6408948 IC50 = 76 nM T59328 C18VEH 6415635 IC50 = 65 nM T59328 C0ITJ4 6419347 IC50 = 4.1 nM T59328 C61JMS 6419746 IC50 = 440000 nM T59328 CZF6Y9 6439072 IC50 = 1000 nM T59328 CO5SZ1 6440837 IC50 > 200 ug.mL-1 T59328 C4KVL5 6441269 IC50 = 19000000 nM T59328 C83XSI 6442618 IC50 = 8 ug.mL-1 T59328 C9YRT1 6447922 IC50 = 4000 nM T59328 CXO27Z 6447923 IC50 = 20000 nM T59328 CTB7N5 6447926 IC50 = 398.11 nM T59328 C49YOE 6447934 IC50 = 3000 nM T59328 CQ3S8L 6450842 IC50 > 100000 nM T59328 C2N0IR 6477203 IC50 > 50000 nM T59328 CL8MC2 6505651 IC50 > 10 ug.mL-1 T59328 CW5YJ2 6536705 IC50 > 100000 nM T59328 C0O8DH 6538899 IC50 = 1680 nM T59328 CUPQ08 6539985 IC50 > 50000 nM T59328 CMEZ23 6540005 IC50 > 50000 nM T59328 CP0XI6 6603792 IC50 = 177 nM T59328 CUJ97R 7023155 IC50 = 6800 nM T59328 C0MGV7 7048595 IC50 = 2800 nM T59328 C14UAT 7574840 IC50 > 10000 nM T59328 CV7L5M 8895911 IC50 > 10000 nM T59328 CY01OB 9209612 IC50 = 57000 nM T59328 CH46ZU 9583801 IC50 > 100000 nM T59328 C4A8RX 9794758 IC50 = 510 nM T59328 C2OL7K 9796455 IC50 = 3700 nM T59328 CZR3M4 9799152 IC50 > 100000 nM T59328 C2B4ZE 9803006 IC50 = 910 nM T59328 CF47BP 9806229 IC50 = 0.79 nM T59328 C72WMK 9808725 IC50 = 91 nM T59328 CZ2MH9 9809611 IC50 = 19 nM T59328 CI3O6X 9814609 IC50 > 100000 nM T59328 CUNV09 9816954 IC50 = 27000 nM T59328 CK2DM9 9818251 IC50 = 100 nM T59328 C4Z2GW 9819930 IC50 = 797 nM T59328 CZ5VX6 9820644 IC50 = 0.2512 nM T59328 CKR04B 9821918 IC50 = 700 nM T59328 CX9DG5 9822042 IC50 > 100000 nM T59328 CRKD07 9825976 IC50 = 33 nM T59328 C1E2DV 9826083 IC50 = 8700 nM T59328 C9TAL6 9826308 IC50 > 48000 nM T59328 C4XU5Z 9828336 IC50 = 27 nM T59328 C5S8FR 9829680 IC50 = 28 nM T59328 CYWI50 9830092 IC50 = 160 nM T59328 CBGE59 9833337 IC50 = 2000 nM T59328 CFPI31 9844683 IC50 = 3200 nM T59328 CSH0A9 9847014 IC50 = 530 nM T59328 CGKC15 9851149 IC50 = 100 nM T59328 C41QWA 9857146 IC50 = 6300 nM T59328 C43FVO 9859850 IC50 = 340 nM T59328 C3UQL7 9860872 IC50 = 100000 nM T59328 C16VXB 9863538 IC50 > 10000 nM T59328 CW8V0K 9864418 IC50 > 25000 nM T59328 CGC0F7 9864462 IC50 = 2.5 nM T59328 CTN7L4 9869773 IC50 = 200 nM T59328 CM5Z8X 9869943 IC50 > 10000 nM T59328 C12PKF 9871380 IC50 = 40 nM T59328 C2FW1X 9872621 IC50 = 18 nM T59328 CS51KJ 9873631 IC50 = 43 nM T59328 CU2N8D 9873657 IC50 = 18 nM T59328 C5NK9U 9873849 IC50 = 27 nM T59328 C5CLD8 9874613 IC50 = 90 nM T59328 CM2QX5 9879615 IC50 = 4100 nM T59328 CSB5D8 9882519 IC50 = 200 nM T59328 CY70OD 9882602 IC50 = 6 nM T59328 CPJ7W2 9882655 IC50 > 20000 nM T59328 CV1A2S 9883384 IC50 = 170 nM T59328 CE47IF 9884465 IC50 = 3 nM T59328 C4R8YV 9884654 IC50 = 1 nM T59328 CUZ07T 9884745 IC50 = 7900 nM T59328 CL5BD2 9885081 IC50 = 39 nM T59328 C2JR8Q 9887521 IC50 = 933.25 nM T59328 CR2B8U 9888491 IC50 = 1704 nM T59328 CXL31W 9890154 IC50 = 2320 nM T59328 CHF7G5 9890746 IC50 > 100000 nM T59328 CIN0E2 9891993 IC50 = 13489.63 nM T59328 CXA5C8 9893493 IC50 = 4200 nM T59328 CE87TX 9893671 IC50 = 24 nM T59328 CEJ05V 9894581 IC50 = 26 nM T59328 C4WQK8 9897300 IC50 = 3.6 nM T59328 CB4DT1 9899125 IC50 = 5600 nM T59328 CP04SA 9906350 IC50 = 10000 nM T59328 C01WSX 9907221 IC50 = 1.6 nM T59328 CO7RU2 9908666 IC50 = 0.4 nM T59328 C2TC1L 9910609 IC50 = 239 nM T59328 C3EUB4 9911005 IC50 > 100000 nM T59328 C9SQU4 9913648 IC50 = 1600 nM T59328 C5GE7T 9917045 IC50 = 5400 nM T59328 CF3KI0 9917474 IC50 = 25 nM T59328 C2DL8U 9927208 IC50 = 4 nM T59328 CYW49X 9927718 IC50 = 10000 nM T59328 CG6A1H 9927800 IC50 > 10000 nM T59328 CWT56C 9930439 IC50 = 86.9 nM T59328 CP2J4W 9930632 IC50 = 3.6 nM T59328 CPYB98 9934935 IC50 = 1910293.07 nM T59328 CU56DE 9937225 IC50 = 23 nM T59328 CLT0U5 9937660 IC50 = 12 nM T59328 CXJR73 9938805 IC50 = 89 nM T59328 CUKH27 9943194 IC50 = 50000 nM T59328 CU78NO 9947433 IC50 > 100000 nM T59328 CYI65J 9948215 IC50 = 29 nM T59328 C6HP3L 9948410 IC50 > 100000 nM T59328 C0U6EJ 9949448 IC50 > 100000 nM T59328 C06JHE 9952784 IC50 = 0.07 nM T59328 CYT7R9 9953676 IC50 > 100000 nM T59328 CI51BV 9954075 IC50 = 645.65 nM T59328 CBE9O6 9954156 IC50 = 36 nM T59328 CJM8R9 9956715 IC50 = 1000 nM T59328 C0ZO2V 9960493 IC50 = 21 nM T59328 CSU19Y 9960734 IC50 = 85 nM T59328 CJ40GO 9965429 IC50 > 100000 nM T59328 CIKN68 9965616 IC50 = 2 ug.mL-1 T59328 CAH50Y 9970231 IC50 = 14100 nM T59328 CM8NB2 9972089 IC50 > 20000 nM T59328 C24MZU 9974694 IC50 = 3.1 nM T59328 CZN09Q 9977010 IC50 > 1000 nM T59328 CCV62S 9978638 IC50 = 1500 nM T59328 CROV41 9979362 IC50 = 850 nM T59328 C6BXQ9 9979953 IC50 = 5000 nM T59328 CA6Z4L 9980337 IC50 = 5000 nM T59328 CFVI29 9981239 IC50 = 8.6 nM T59328 CB2KF5 9981727 IC50 = 35 nM T59328 C37GXK 9983303 IC50 > 25000 nM T59328 CH03DY 9984664 IC50 = 10320 nM T59328 C29SOH 9985870 IC50 > 100000 nM T59328 CQZF34 9994794 IC50 > 100000 nM T59328 CO4N3Q 9995374 IC50 > 100000 nM T59328 CFG0E8 9996177 IC50 = 20000 nM T59328 CF0SE3 9998325 IC50 = 900 nM T59328 CMYI47 10002824 IC50 = 2 nM T59328 CNY2F1 10005402 IC50 = 2 nM T59328 C26QHZ 10005638 IC50 > 10000 nM T59328 CQX39R 10006530 IC50 = 80 nM T59328 C0EWK9 10007087 IC50 = 10000 nM T59328 CH7DN2 10009462 IC50 = 16900 nM T59328 CF2V4B 10016116 IC50 > 10000 nM T59328 C7WJ5H 10016952 IC50 = 66100 nM T59328 CWH02V 10018196 IC50 > 20000 nM T59328 CA5E4R 10019589 IC50 = 1000 nM T59328 C86HYI 10020830 IC50 = 70 nM T59328 C53UTR 10022185 IC50 = 8800 nM T59328 C1Y0PX 10023383 IC50 < 5 nM T59328 CO2PA9 10029703 IC50 = 5390 nM T59328 C19XDW 10032479 IC50 > 100000 nM T59328 C0IA4P 10037831 IC50 = 8700 nM T59328 CXL0R8 10038606 IC50 > 100000 nM T59328 CD4Z1B 10040645 IC50 = 9500 nM T59328 C8TY1B 10040646 IC50 = 3000 nM T59328 C2M8VJ 10040715 IC50 > 20000 nM T59328 C8VNJ1 10041429 IC50 = 37500 nM T59328 C0XAV7 10041970 IC50 = 3000 nM T59328 CE98SN 10041980 IC50 > 20000 nM T59328 C1YV0B 10043236 IC50 = 100 nM T59328 C8IS1F 10043899 IC50 = 400 nM T59328 C25JLD 10043994 IC50 = 2000 nM T59328 CF03ZB 10044469 IC50 = 90 nM T59328 CAZ71W 10045755 IC50 ~ 4000 nM T59328 CJ6L3T 10046873 IC50 > 50000 nM T59328 CG57EC 10047098 IC50 = 300 nM T59328 C7YD1X 10048045 IC50 > 25000 nM T59328 C54AEL 10048519 IC50 = 2100 nM T59328 C9VQZ3 10053637 IC50 = 47000 nM T59328 CFS2H4 10053638 IC50 > 100000 nM T59328 C32WOU 10058766 IC50 > 20000 nM T59328 C6K0XB 10064040 IC50 = 670 nM T59328 CR7TY8 10064290 IC50 > 20000 nM T59328 C5UPR6 10065338 IC50 = 6.4 nM T59328 CBF54I 10066030 IC50 = 8700 nM T59328 C82XJV 10067396 IC50 = 80 nM T59328 CH2WO5 10067548 IC50 = 490 nM T59328 C2L3JB 10068026 IC50 = 6900 nM T59328 C0DR5I 10068517 IC50 = 0.6761 nM T59328 C7DNB8 10070557 IC50 = 21 nM T59328 CCK25W 10070969 IC50 = 45800 nM T59328 CK8RL4 10071409 IC50 = 125 ug.mL-1 T59328 C7J8YN 10073101 IC50 = 8800 nM T59328 C1JUF8 10073832 IC50 > 10000 nM T59328 CF1D6Y 10075240 IC50 > 10000 nM T59328 CC0J9E 10075664 IC50 = 25 nM T59328 CD5B6O 10076837 IC50 > 100000 nM T59328 CMK64J 10084671 IC50 = 21000 nM T59328 C8A1TH 10085171 IC50 > 100000 nM T59328 CM96YH 10085557 IC50 = 600 nM T59328 C2C1BP 10089048 IC50 > 25000 nM T59328 C8HEJ2 10092460 IC50 = 800 nM T59328 COW60X 10092803 IC50 = 400 nM T59328 CX6N2G 10092804 IC50 = 360 nM T59328 CH62FG 10093300 IC50 = 7000 nM T59328 CF09NK 10098235 IC50 = 3830 nM T59328 CK50LJ 10100761 IC50 = 47000 nM T59328 C10SZX 10106602 IC50 > 20000 nM T59328 CZ9Y1G 10106867 IC50 = 11 nM T59328 C3P8WK 10110378 IC50 > 100000 nM T59328 C63CFD 10111108 IC50 > 100000 nM T59328 C7TA9J 10113568 IC50 = 10000 nM T59328 C5SV9C 10114464 IC50 = 64 nM T59328 C80ZDK 10115240 IC50 = 90 nM T59328 C7C1IG 10116123 IC50 = 110 nM T59328 CMK79O 10117051 IC50 = 200 nM T59328 CYV4I1 10127271 IC50 = 9300 nM T59328 CA31MX 10131256 IC50 = 650 nM T59328 CV4QA0 10136035 IC50 = 4800 nM T59328 C53JSE 10136105 IC50 = 680 nM T59328 CL42XS 10136330 IC50 > 100000 nM T59328 CREM37 10151881 IC50 = 35 nM T59328 CC4X6M 10152238 IC50 = 5 nM T59328 C5HB2P 10152514 IC50 = 48 nM T59328 C14ZEP 10156890 IC50 = 1061 nM T59328 CUW34X 10157645 IC50 = 100000 nM T59328 CUD7L1 10159833 IC50 = 45 nM T59328 CZE4S6 10159951 IC50 = 10 nM T59328 CA40TZ 10161969 IC50 = 790 nM T59328 CHU9C6 10162630 IC50 = 690 nM T59328 CK4OH0 10162954 IC50 = 698 nM T59328 CGW26V 10163178 IC50 = 0.5 nM T59328 C9LH1R 10172616 IC50 = 720 nM T59328 CZ4X7O 10172837 IC50 > 10000 nM T59328 CC56EH 10173248 IC50 = 10 nM T59328 CC78NE 10179293 IC50 = 853 nM T59328 C6H3FI 10180188 IC50 = 21 nM T59328 COC30E 10181160 IC50 > 100000 nM T59328 C3GFB0 10194325 IC50 = 55 nM T59328 CNYA34 10194617 IC50 = 9000 nM T59328 CQP8Y1 10194801 IC50 = 90 nM T59328 CI4Q0J 10195479 IC50 = 73 nM T59328 C1TX8D 10198953 IC50 = 29400 nM T59328 C2RLF5 10199254 IC50 = 200 nM T59328 C47FXG 10200918 IC50 = 1139 nM T59328 CGOT91 10207821 IC50 > 100000 nM T59328 C5YCN2 10215023 IC50 > 100000 nM T59328 CZ0XD7 10215809 IC50 = 390 nM T59328 CP81YE 10216042 IC50 = 2 nM T59328 CVQ53X 10216257 IC50 = 560 nM T59328 C36YTW 10216482 IC50 = 45 nM T59328 CZ2A0F 10216910 IC50 = 5 nM T59328 CNTU23 10217083 IC50 = 60 nM T59328 CSGL59 10217304 IC50 = 170 nM T59328 CEW30I 10217590 IC50 = 61 nM T59328 C74AGX 10222656 IC50 = 71 nM T59328 C67POS 10223065 IC50 = 1620 nM T59328 CCVU79 10226418 IC50 = 160 nM T59328 C2KSD3 10227095 IC50 = 350 nM T59328 C6QP4E 10227907 IC50 = 63 nM T59328 CD7J3O 10231458 IC50 > 30000 nM T59328 CPD6Z9 10236164 IC50 > 100000 nM T59328 CV7PU8 10237247 IC50 = 85 nM T59328 C0UN1C 10245626 IC50 > 20000 nM T59328 CQ3LT1 10245856 IC50 = 14 nM T59328 CSGD16 10246246 IC50 > 7000 nM T59328 CYMD04 10246609 IC50 > 20000 nM T59328 CLV83M 10246831 IC50 > 50000 nM T59328 CU53QW 10247949 IC50 = 5000 nM T59328 CGME21 10248155 IC50 > 100000 nM T59328 C97GRN 10248747 IC50 = 100000 nM T59328 CNH85V 10249869 IC50 = 1300 nM T59328 CC9E5Q 10249989 IC50 > 10000 nM T59328 C1WL8B 10251852 IC50 = 22800 nM T59328 CH30RC 10253133 IC50 > 10000 nM T59328 C1UB5A 10253204 IC50 = 309.03 nM T59328 C32KTH 10253992 IC50 = 21200 nM T59328 CG2TF7 10255849 IC50 = 7700 nM T59328 CBR9P3 10257058 IC50 = 17500 nM T59328 C6G8NR 10264200 IC50 > 100000 nM T59328 C3HF6S 10264201 IC50 > 100000 nM T59328 CBI47E 10264222 IC50 > 100000 nM T59328 CF81EM 10265006 IC50 > 100000 nM T59328 CHFZ23 10266516 IC50 = 180 nM T59328 CWY4U3 10267270 IC50 = 460 nM T59328 CJGH26 10275985 IC50 = 2290 nM T59328 C6PL7V 10276061 IC50 = 64 nM T59328 CY67TW 10287149 IC50 = 11 nM T59328 C4W6JL 10287402 IC50 = 18 nM T59328 CT3W9O 10287552 IC50 = 2 nM T59328 CE7Q8U 10288283 IC50 = 8 nM T59328 C9K0SA 10288761 IC50 = 140 nM T59328 CJ4D9B 10288917 IC50 = 240 nM T59328 CNU74Z 10288918 IC50 = 780 nM T59328 CCE64Z 10288920 IC50 = 35 nM T59328 CN51JQ 10292737 IC50 > 100000 nM T59328 C3FL9K 10295633 IC50 = 4400 nM T59328 C8NMA6 10295839 IC50 = 810 nM T59328 C7SFI1 10296883 IC50 > 10000 nM T59328 CVO54Z 10300451 IC50 = 40 nM T59328 C8RD3V 10301884 IC50 = 900 nM T59328 C1AKH9 10303277 IC50 > 1000 nM T59328 CY0A3T 10309300 IC50 = 3 nM T59328 C8DQ9O 10309491 IC50 = 1100 nM T59328 C3MJB0 10309561 IC50 = 11 nM T59328 CGF21D 10310843 IC50 = 68 nM T59328 C0SY1J 10314618 IC50 > 20000 nM T59328 CD34UM 10317124 IC50 = 2500 nM T59328 CW85MK 10317696 IC50 = 4000 nM T59328 CM1X0V 10318022 IC50 = 174 nM T59328 C39YNC 10318148 IC50 > 100000 nM T59328 C1KFM8 10318154 IC50 = 230 nM T59328 CK83IU 10318851 IC50 = 110 nM T59328 C27CDR 10319118 IC50 = 7300 nM T59328 CUC58I 10320940 IC50 = 0.12 nM T59328 CEN48D 10322889 IC50 = 790 nM T59328 CN23SU 10324074 IC50 > 1000 nM T59328 C6WJB8 10325906 IC50 > 50000 nM T59328 CCK42E 10327195 IC50 = 5300 nM T59328 CX7NM0 10327196 IC50 > 100000 nM T59328 CQ03XB 10327197 IC50 > 100000 nM T59328 COB74A 10330538 IC50 > 20000 nM T59328 CG1AS6 10333483 IC50 = 20000 nM T59328 COC7P1 10333957 IC50 > 100000 nM T59328 CQ80HY 10337047 IC50 = 1100 nM T59328 CET21U 10337153 IC50 = 1100 nM T59328 C9GK3M 10342546 IC50 = 1000 nM T59328 CU8LT7 10345125 IC50 > 50000 nM T59328 CD2H0G 10347728 IC50 = 43000 nM T59328 CNJ97S 10348925 IC50 = 5500 nM T59328 CZ0UL8 10349829 IC50 = 13000 nM T59328 CYCM39 10355659 IC50 > 100000 nM T59328 C37AMD 10356450 IC50 > 100000 nM T59328 C4DOQ9 10356451 IC50 = 7800 nM T59328 CE08LX 10356808 IC50 = 6000 nM T59328 CYI4N2 10357604 IC50 = 400 nM T59328 CT19AL 10359253 IC50 = 27500 nM T59328 C19VUI 10360971 IC50 > 50000 nM T59328 C3L5UZ 10361853 IC50 > 50000 nM T59328 C8RW0D 10362209 IC50 = 20 nM T59328 CD1R3L 10362325 IC50 = 200 nM T59328 C8H1OJ 10371203 IC50 = 1700 nM T59328 C7ACN5 10383837 IC50 = 700 nM T59328 CVP85S 10385997 IC50 = 10000 nM T59328 C6ZF0X 10386217 IC50 > 100000 nM T59328 C36GIL 10386874 IC50 = 4700 nM T59328 CQB9H7 10389422 IC50 = 4800 nM T59328 CA8B5T 10390073 IC50 = 1100 nM T59328 CQIK61 10406106 IC50 = 900 nM T59328 CF74ID 10406267 IC50 = 2500 nM T59328 CBMW34 10406907 IC50 > 20000 nM T59328 C34JQT 10407176 IC50 > 100000 nM T59328 C4SGL2 10407341 IC50 > 100000 nM T59328 CC13FP 10408738 IC50 = 90 nM T59328 C9RCU7 10408993 IC50 = 470 nM T59328 C4PV3R 10409198 IC50 = 5600 nM T59328 C32REN 10411907 IC50 = 4 nM T59328 CFJ2S1 10413621 IC50 >> 5000 nM T59328 CHPR58 10416818 IC50 = 12000 nM T59328 CVK10W 10421743 IC50 > 20000 nM T59328 CP6N2J 10423146 IC50 > 100000 nM T59328 C4T5WG 10424297 IC50 = 400 nM T59328 CHID58 10425395 IC50 > 20000 nM T59328 CQ43JU 10426229 IC50 = 400 nM T59328 CQR85O 10427421 IC50 > 20000 nM T59328 C7HBP6 10429593 IC50 > 10000 nM T59328 CE6P0T 10429844 IC50 = 50 nM T59328 C2SXE3 10430383 IC50 = 1000 nM T59328 CP14EC 10430484 IC50 = 3400 nM T59328 C3MI7D 10430804 IC50 = 300 nM T59328 CFLH53 10432113 IC50 = 800 nM T59328 C56SVY 10434122 IC50 = 1250 nM T59328 CN5BF4 10434923 IC50 = 50000 nM T59328 C7QU9X 10437879 IC50 > 100000 nM T59328 CXA85V 10439212 IC50 = 6100 nM T59328 CQHS12 10445612 IC50 > 25000 nM T59328 CEU25H 10445729 IC50 > 100000 nM T59328 C9XLN7 10446123 IC50 = 5400 nM T59328 C3LY4K 10447743 IC50 = 300 nM T59328 CUX75O 10450005 IC50 > 50000 nM T59328 CT42KE 10450849 IC50 > 100000 nM T59328 CL7PF2 10451087 IC50 = 3400 nM T59328 C9GJZ5 10453233 IC50 = 1000 nM T59328 CZ09AI 10454066 IC50 = 2700 nM T59328 CSZ40F 10455755 IC50 = 1250 nM T59328 C95LYF 10457505 IC50 > 100000 nM T59328 CYF3P4 10468511 IC50 = 9000 nM T59328 CW23SQ 10468973 IC50 > 100000 nM T59328 C2CVB8 10470221 IC50 > 100000 nM T59328 C4DTZ5 10470384 IC50 > 20000 nM T59328 CH4CY9 10471016 IC50 = 700 nM T59328 CI7BO0 10471069 IC50 = 7000 nM T59328 C3JIZ2 10473386 IC50 > 20000 nM T59328 CC5OM4 10473589 IC50 > 200 ug.mL-1 T59328 C5PAU6 10475547 IC50 = 100000 nM T59328 CC98AG 10475666 IC50 = 3000 nM T59328 C1GKT0 10476486 IC50 = 1000 nM T59328 CZ45NX 10476762 IC50 > 100000 nM T59328 CR07PO 10477008 IC50 = 700 nM T59328 CM9F3D 10477397 IC50 > 1000 nM T59328 C7PLI5 10478569 IC50 > 10000 nM T59328 CRX6F0 10479082 IC50 > 25000 nM T59328 COW2Q5 10483554 IC50 > 100000 nM T59328 CD7XE3 10484487 IC50 > 100000 nM T59328 CJWH60 10489322 IC50 > 100000 nM T59328 C0EV8B 10494548 IC50 = 6000 nM T59328 C05ANY 10494804 IC50 = 538 nM T59328 CZ06SL 10495153 IC50 > 100000 nM T59328 C8DH5W 10499619 IC50 = 12500 nM T59328 C78FPR 10501266 IC50 = 1800 nM T59328 C1O6YQ 10502559 IC50 > 50000 nM T59328 CB76HG 10504176 IC50 = 2 nM T59328 C3DK8I 10520057 IC50 = 0.25 nM T59328 CB3MW7 10522352 IC50 = 0.91 nM T59328 C7RFN2 10523147 IC50 = 1.1 nM T59328 CLH12I 10523411 IC50 = 291 nM T59328 C0GP2I 10523766 IC50 > 5000 nM T59328 C38RSF 10528818 IC50 = 0.16 nM T59328 CBC2E1 10530118 IC50 = 3 nM T59328 C5SVT4 10537949 IC50 > 100000 nM T59328 CU0E9F 10538285 IC50 = 6920 nM T59328 C3VPC7 10538965 IC50 > 100000 nM T59328 CG63KU 10539833 IC50 = 1200 nM T59328 CXT20A 10541248 IC50 = 500 nM T59328 C8VJX1 10542530 IC50 > 5000 nM T59328 C7JX3G 10547930 IC50 = 4.8 nM T59328 CP64DQ 10549169 IC50 > 5000 nM T59328 CSG53A 10549915 IC50 = 377 nM T59328 CXFB12 10555151 IC50 = 7000 nM T59328 CGAW17 10562306 IC50 > 100000 nM T59328 C6AJI9 10562777 IC50 > 100000 nM T59328 C95SZN 10564143 IC50 = 58800 nM T59328 CR91ZK 10564707 IC50 = 420 nM T59328 CW16DN 10568777 IC50 = 10 nM T59328 CX67AG 10569366 IC50 = 46 nM T59328 CE5L6D 10587839 IC50 > 100000 nM T59328 C1ICU3 10589889 IC50 = 860 nM T59328 CP8J4O 10590515 IC50 = 1270 nM T59328 CM8N6L 10593765 IC50 > 100000 nM T59328 C64CRU 10599506 IC50 > 10000 nM T59328 CF8IH9 10600888 IC50 = 3.9 nM T59328 COB2X8 10602350 IC50 = 7000 nM T59328 CY51ET 10611103 IC50 > 10000 nM T59328 CI30LZ 10613858 IC50 > 100000 nM T59328 CTG7H5 10614224 IC50 = 7830 nM T59328 C0LHE5 10615400 IC50 = 25 nM T59328 CWU4L7 10616703 IC50 = 10000 nM T59328 CNE92Q 10616753 IC50 = 230 nM T59328 CX8R0T 10618464 IC50 = 5400 nM T59328 CZ5L3U 10635276 IC50 = 200 nM T59328 CH6Z3L 10635478 IC50 > 100000 nM T59328 CB97UD 10636005 IC50 > 100000 nM T59328 C0C8QK 10638407 IC50 = 170 nM T59328 C1JY5N 10638517 IC50 = 25700 nM T59328 CG93BK 10640018 IC50 > 10000 nM T59328 C2UWA0 10658651 IC50 > 100000 nM T59328 CZ78VR 10660240 IC50 = 820 nM T59328 CZ40OF 10660724 IC50 > 5000 nM T59328 C64DFG 10662351 IC50 = 0.48 nM T59328 C5L0IX 10663368 IC50 > 100000 nM T59328 C9Z7XH 10663503 IC50 > 100000 nM T59328 C5M0HJ 10670094 IC50 = 45 nM T59328 CKA30X 10671481 IC50 = 0.51 nM T59328 CFGL61 10672994 IC50 = 6.6 nM T59328 CDV84T 10673774 IC50 = 1.8 nM T59328 CR9N8Z 10674806 IC50 > 100000 nM T59328 CH1G6P 10682457 IC50 = 44000 nM T59328 CLQP93 10683468 IC50 > 20000 nM T59328 CAVX96 10686149 IC50 > 100000 nM T59328 C51VNS 10691590 IC50 = 0.69 nM T59328 C6BK7Q 10691652 IC50 = 2.1 nM T59328 CK85TP 10692159 IC50 = 3000 nM T59328 C0AOG5 10696486 IC50 = 21 nM T59328 C7INC2 10706114 IC50 = 1250 nM T59328 CU6G5Y 10708835 IC50 > 100000 nM T59328 C54UAK 10728035 IC50 > 100000 nM T59328 CZVK65 10729749 IC50 = 550 nM T59328 CJO8Q1 10738332 IC50 = 1360 nM T59328 CN8GS6 10738988 IC50 = 1.2 nM T59328 CVX5L1 10742427 IC50 = 27 nM T59328 CXSH91 10753550 IC50 > 100000 nM T59328 C25MWP 10754509 IC50 > 10000 nM T59328 CVPW04 10755069 IC50 > 100000 nM T59328 CYAL86 10759828 IC50 = 3.3 nM T59328 CVO13S 10759989 IC50 = 41000 nM T59328 CD26KN 10760134 IC50 > 5000 nM T59328 CL0XH6 10762274 IC50 = 8000 nM T59328 CQO0A2 10762478 IC50 > 5000 nM T59328 C3WR0Q 10779668 IC50 > 100000 nM T59328 C7YJ4L 10782259 IC50 = 1.6 nM T59328 CF5T1H 10783444 IC50 = 19300 nM T59328 CFK51I 10784704 IC50 > 5000 nM T59328 C71QOK 10789593 IC50 = 1.5 nM T59328 C62FWK 10791534 IC50 = 88 nM T59328 C1OXH6 10803234 IC50 = 8 nM T59328 CT7O1G 10803426 IC50 = 10000 nM T59328 CH7Q9F 10804454 IC50 = 14000 nM T59328 C3QT8I 10806455 IC50 = 360 nM T59328 CNC84J 10811119 IC50 > 10000 nM T59328 CK0W6X 10815675 IC50 = 0.78 nM T59328 C89PRO 10826146 IC50 = 2500 nM T59328 CRJM76 10826740 IC50 = 16300 nM T59328 CDP61C 10832923 IC50 = 108 nM T59328 C3TCG9 10834960 IC50 > 5000 nM T59328 CWX4V1 10838598 IC50 = 2.7 nM T59328 CYPB29 10841700 IC50 = 6.7 ug.mL-1 T59328 C18MDA 10848423 IC50 = 570 nM T59328 C49OYX 10850623 IC50 > 10000 nM T59328 C01KXI 10854884 IC50 = 0.75 nM T59328 CGFO65 10856252 IC50 > 20000 nM T59328 C9QG7J 10868706 IC50 = 8400 nM T59328 C8IZ4B 10870494 IC50 = 24 nM T59328 CI5FC1 10875157 IC50 = 100000 nM T59328 C67ZFI 10880751 IC50 = 29 nM T59328 CTI84S 10884588 IC50 = 960 nM T59328 C7DK8H 10885120 IC50 = 2700 nM T59328 CA8J0B 10902421 IC50 = 335 nM T59328 CT7CA1 10905749 IC50 = 38 nM T59328 CJ4P5T 10905857 IC50 > 100000 nM T59328 CP5XT0 10906920 IC50 = 89.13 nM T59328 CBM57K 10918242 IC50 = 10471.29 nM T59328 CF9O7M 10926736 IC50 = 9300 nM T59328 CIRP84 10928765 IC50 = 5220 nM T59328 C60QTH 10938977 IC50 = 238 nM T59328 CI01XA 10951285 IC50 = 2640 nM T59328 CEKW21 10972694 IC50 = 560 nM T59328 C1I6VX 10973080 IC50 = 4840 nM T59328 CTY19K 10973186 IC50 = 250 nM T59328 COE13S 10983483 IC50 = 2290 nM T59328 C90YUA 10992313 IC50 = 11 nM T59328 C2AK4W 11005320 IC50 = 930 nM T59328 C3OM5X 11012217 IC50 = 13350 nM T59328 C0Y5PH 11016075 IC50 = 330 nM T59328 CM4JD2 11037303 IC50 = 7500 nM T59328 CJ05CL 11048367 IC50 > 30000 nM T59328 C9QI8E 11055442 IC50 = 8000 nM T59328 C2FPI5 11071370 IC50 = 150 nM T59328 C3UTD8 11080556 IC50 = 25 nM T59328 CR91TM 11102890 IC50 = 2880 nM T59328 C8TA4Z 11129889 IC50 > 100000 nM T59328 CR2O3F 11155047 IC50 > 10000 nM T59328 COB20T 11157041 IC50 = 768 nM T59328 CUIX38 11157794 IC50 = 30 nM T59328 C2W5OA 11165103 IC50 = 6900 nM T59328 C0VD5M 11168387 IC50 = 345 nM T59328 CSZ6B2 11168731 IC50 = 650 nM T59328 CQ7PU5 11178756 IC50 = 36 nM T59328 C7XU5W 11180271 IC50 = 24 nM T59328 C9Z6AG 11180494 IC50 = 500 nM T59328 CHV1P9 11180599 IC50 = 250 nM T59328 C2B7HJ 11180905 IC50 = 31 nM T59328 CUVW02 11186266 IC50 = 7500 nM T59328 CRG7B6 11192261 IC50 = 277 nM T59328 CA6L9Y 11192678 IC50 = 20 nM T59328 C2PMR9 11192753 IC50 = 15 nM T59328 CA07YO 11193143 IC50 = 574 nM T59328 CABZ27 11197585 IC50 = 7000 nM T59328 CQG17S 11202074 IC50 = 1020 nM T59328 C0K8NB 11202869 IC50 = 770 nM T59328 C16HXD 11203436 IC50 = 45 nM T59328 C7H8AD 11203663 IC50 = 42 nM T59328 C87QSN 11203886 IC50 = 100 nM T59328 C2NUG6 11210620 IC50 = 1000 nM T59328 C1YB7C 11220978 IC50 = 40 nM T59328 CNZ2H8 11226874 IC50 = 770 nM T59328 CMZ8S5 11227115 IC50 = 11 nM T59328 C4HUM2 11232168 IC50 = 250 nM T59328 CIJG62 11232492 IC50 = 8900 nM T59328 CH7D3X 11233762 IC50 > 100000 nM T59328 CD43EZ 11234126 IC50 = 900 nM T59328 C2W5RC 11235063 IC50 > 50000 nM T59328 C98HRX 11237508 IC50 = 185 nM T59328 CXN98V 11238293 IC50 = 341 nM T59328 CSX6P5 11238512 IC50 = 34 nM T59328 CWOU43 11238694 IC50 = 110 nM T59328 CG07FL 11238864 IC50 = 360 nM T59328 C0QN4V 11238875 IC50 = 343 nM T59328 COI7A0 11245620 IC50 = 10000 nM T59328 CU27LB 11246488 IC50 = 0.66 nM T59328 CGP6U2 11249521 IC50 = 1191 nM T59328 CO97YK 11249776 IC50 = 23 nM T59328 CJ02WR 11249881 IC50 = 223 nM T59328 CWF87N 11260603 IC50 = 372 nM T59328 CNBX16 11270660 IC50 = 2730 nM T59328 CR35NY 11273032 IC50 = 28 nM T59328 CO2E3W 11280238 IC50 > 50000 nM T59328 CUO27S 11282791 IC50 > 500 nM T59328 C5EO4X 11284905 IC50 = 34 nM T59328 CJ6R3N 11284937 IC50 = 65 nM T59328 CIV3Y6 11285080 IC50 = 282 nM T59328 C8FGR1 11288910 IC50 = 3250 nM T59328 CI63ZB 11291617 IC50 = 3400 nM T59328 CBOP58 11293798 Ki > 10000 nM T59328 C0HM3D 11293802 IC50 = 1000 nM T59328 CH02JX 11296170 IC50 = 195 nM T59328 C5Z6NC 11296256 IC50 = 163 nM T59328 CU9ER4 11296411 IC50 = 238 nM T59328 CG7VP5 11302688 IC50 = 5800 nM T59328 C84VYL 11303451 IC50 = 10 nM T59328 C6ZF7L 11303620 IC50 = 6000 nM T59328 CP3BM8 11307161 IC50 = 12700 nM T59328 C18BHK 11307255 IC50 = 445 nM T59328 C64SCF 11307581 IC50 = 32 nM T59328 C6OQC2 11307602 IC50 = 26 nM T59328 CZN3Q6 11307866 IC50 = 82 nM T59328 CANY24 11311217 IC50 = 100000 nM T59328 C0SO6D 11312797 IC50 = 412.8 nM T59328 CRD9E5 11314043 IC50 = 45000 nM T59328 CR9E2X 11316711 IC50 = 6.4 nM T59328 CLX54H 11317348 IC50 > 10000 nM T59328 CRN20W 11326156 IC50 = 37 nM T59328 C2TP7E 11327841 IC50 = 6300 nM T59328 CM48NO 11336573 IC50 = 2000 nM T59328 CKY3E2 11338122 IC50 > 50000 nM T59328 CF3W8U 11338513 IC50 = 1900 nM T59328 CSZ8P5 11340298 IC50 = 250 nM T59328 CT7CG8 11341400 IC50 = 13000 nM T59328 CXI48D 11342107 IC50 = 165 nM T59328 C8FQY5 11342284 IC50 = 31 nM T59328 CO2E6V 11342331 IC50 = 7 nM T59328 CLA1W0 11342405 IC50 = 75 nM T59328 C3KC4P 11353443 IC50 = 53 nM T59328 C49AZU 11354013 IC50 = 16 nM T59328 CDZR14 11357877 IC50 = 100 nM T59328 C0J2TB 11359024 IC50 = 50 nM T59328 C26BZX 11362471 Ki > 10000 nM T59328 CK14GM 11365122 IC50 = 111 nM T59328 C5WI2V 11365297 IC50 = 20 nM T59328 CX5FE9 11365342 IC50 = 51 nM T59328 CYF58P 11365726 IC50 = 125 nM T59328 C3OCV2 11371778 IC50 = 7100 nM T59328 C43NPS 11373886 IC50 = 30 nM T59328 CN4O0Q 11376079 IC50 = 894 nM T59328 CT3W2J 11376208 IC50 = 100 nM T59328 C4H0ZP 11380375 IC50 = 150 nM T59328 C10XFS 11382411 IC50 = 10 nM T59328 C3WYU1 11387244 IC50 = 340 nM T59328 CWXB93 11397177 Ki > 10000 nM T59328 CA9N1G 11398437 IC50 = 519 nM T59328 CN4WA3 11398461 IC50 = 130 nM T59328 CBV84Q 11398999 IC50 = 64 nM T59328 C2V7RQ 11399289 IC50 = 10 nM T59328 CY76XJ 11399310 IC50 = 214 nM T59328 C6UXH4 11399331 IC50 = 188 nM T59328 CV2IN9 11404920 IC50 = 25 nM T59328 CX25IH 11407794 IC50 = 365 nM T59328 CV5IR8 11410608 IC50 = 24 nM T59328 C9N3PO 11410634 IC50 = 400 nM T59328 CG7ES9 11410940 IC50 = 221 nM T59328 C15VAK 11420132 IC50 = 250 nM T59328 C94QJA 11420204 IC50 = 7 nM T59328 C1I4JO 11421443 IC50 = 41 nM T59328 CTCG60 11421783 IC50 = 401 nM T59328 CU6FD4 11421877 IC50 = 380 nM T59328 C0APW4 11422034 IC50 > 10000 nM T59328 C0KWX9 11422340 IC50 = 98 nM T59328 C5KWS9 11422548 IC50 = 321 nM T59328 C7AI2V 11432911 IC50 > 25000 nM T59328 C3EXM4 11440028 IC50 > 50000 nM T59328 CYD2A6 11440253 IC50 = 10 nM T59328 C3PFX4 11444623 IC50 = 78 nM T59328 CXV39N 11444862 IC50 = 362 nM T59328 CQ27HA 11452941 IC50 = 2000 nM T59328 CWI62M 11454712 IC50 = 35 nM T59328 C4LZ0F 11455794 IC50 = 285 nM T59328 CFHP63 11456360 IC50 = 990 nM T59328 C7I6AG 11474111 IC50 > 100000 nM T59328 C6M9NC 11477626 IC50 = 5500 nM T59328 CD8RQ7 11478340 IC50 = 403 nM T59328 CVFE14 11478925 IC50 = 68 nM T59328 CA0E8N 11484663 IC50 = 1100 nM T59328 C5O2TE 11486373 IC50 = 1000 nM T59328 C62KHL 11489786 IC50 = 45 nM T59328 CG7XZ1 11490270 IC50 = 63 nM T59328 CKU96Z 11490477 IC50 = 1569 nM T59328 CZI6D9 11493632 IC50 = 10000 nM T59328 C0H6QS 11495680 IC50 = 55 nM T59328 C6-AUG 11496207 IC50 = 44 nM T59328 C40GHQ 11502866 IC50 = 79 nM T59328 CIW9L5 11502867 IC50 = 10 nM T59328 CLWG73 11502887 IC50 = 74 nM T59328 C08APU 11503073 IC50 = 31 nM T59328 C2JD4P 11509595 IC50 = 10.08 nM T59328 CK2Q0X 11516978 IC50 = 120 nM T59328 CR0M9S 11517095 IC50 = 918 nM T59328 CH2IZ9 11517688 IC50 = 5200 nM T59328 CU13WV 11518389 IC50 = 0.5 nM T59328 C91JCX 11518627 IC50 = 8 nM T59328 CF0YW7 11518637 IC50 = 11 nM T59328 CV3NK7 11524106 IC50 = 4.5 nM T59328 CQ63ER 11524582 IC50 = 31.62 nM T59328 C5V7WY 11525136 IC50 = 21700 nM T59328 CI5ET2 11525434 IC50 = 21 nM T59328 CPE53F 11526238 IC50 = 6 nM T59328 C7HMO6 11526786 IC50 > 10000 nM T59328 CL7X4Q 11530963 IC50 = 32000 nM T59328 C5BM4T 11531799 IC50 = 9 nM T59328 C53OSD 11532048 IC50 = 40 nM T59328 CT75DZ 11532242 IC50 = 4.5 nM T59328 CC4QM5 11532676 IC50 = 20 nM T59328 CY6L8I 11532718 IC50 > 10000 nM T59328 C1SGF3 11533556 IC50 = 14 nM T59328 CSKF56 11538667 IC50 = 19.1 nM T59328 CTG83F 11539329 Ki > 1800 nM T59328 C5VO2C 11539461 IC50 = 3.1 nM T59328 C4SNI6 11542889 IC50 > 10000 nM T59328 CGN83M 11544306 IC50 = 10000 nM T59328 C01FVM 11546457 IC50 = 20 nM T59328 CLBH14 11547991 IC50 = 9 nM T59328 C37WYM 11552033 IC50 = 10.9 nM T59328 C7WO0I 11552307 IC50 = 16 nM T59328 C23INE 11552309 IC50 = 9.31 nM T59328 CX6KD1 11553647 IC50 = 6.8 nM T59328 CPT4K5 11554463 IC50 = 294 nM T59328 C3MD0B 11557040 IC50 = 5 nM T59328 CI50OC 11558284 IC50 = 4 nM T59328 C2DM7W 11560794 IC50 = 19300 nM T59328 CB46CA 11561058 IC50 = 77 nM T59328 CS2U5G 11561468 IC50 = 33 nM T59328 CZ9N6O 11561637 IC50 = 30700 nM T59328 CXT51U 11561779 IC50 = 8 nM T59328 CACS26 11561968 Ki > 2000 nM T59328 CNBM81 11562171 IC50 = 9 nM T59328 CKUR82 11568720 IC50 = 1.3 nM T59328 CNV08X 11569158 IC50 = 22 nM T59328 CZ1H0X 11569258 IC50 = 2800 nM T59328 C2R0XV 11569434 IC50 = 104 nM T59328 CO8UB2 11569903 IC50 = 327 nM T59328 COGM15 11574917 IC50 = 1000 nM T59328 CI4P0T 11575228 IC50 = 27000 nM T59328 CU3Q1T 11576231 IC50 = 40 nM T59328 CA74QZ 11581908 IC50 = 5010 nM T59328 CM8NI3 11582856 IC50 = 45900 nM T59328 CW5ZP3 11583431 IC50 > 100000 nM T59328 CO9KP5 11583459 IC50 = 9600 nM T59328 CXMY21 11583563 IC50 = 76 nM T59328 C8ZHL0 11589515 IC50 = 67 nM T59328 C8E5DA 11589674 IC50 > 10000 nM T59328 CMIL86 11590363 Ki > 1800 nM T59328 CN31OR 11590557 IC50 = 1.7 nM T59328 CCPK51 11590799 IC50 = 32 nM T59328 CK4E6V 11591222 IC50 = 2000 nM T59328 CR06MA 11595844 IC50 = 1.4 nM T59328 CE6P8L 11595868 IC50 = 10000 nM T59328 C0NV9Y 11596881 IC50 = 8 nM T59328 CHZ38O 11597061 IC50 = 17 nM T59328 CP1O4N 11597180 IC50 = 17 nM T59328 CR1FG0 11604864 IC50 = 4.3 nM T59328 CC48BK 11605761 IC50 = 60 nM T59328 CFEK68 11606101 IC50 = 3 nM T59328 CF7P3R 11611500 IC50 = 18 nM T59328 C85QTY 11611655 IC50 = 1500 nM T59328 C7TA0C 11612021 IC50 = 42 nM T59328 C9T3VC 11613187 IC50 = 2.7 nM T59328 CSKW87 11617204 IC50 = 240 nM T59328 CEO7I2 11618876 IC50 = 8.95 nM T59328 CZJU74 11619195 IC50 = 5900 nM T59328 C7SFP9 11619763 IC50 = 333 nM T59328 CO68CD 11619972 IC50 = 1 nM T59328 C1BLZ5 11620055 IC50 = 9 nM T59328 C5B3XJ 11620410 IC50 > 25000 nM T59328 CJ6NA8 11620487 IC50 < 1 nM T59328 C5KHN0 11625514 IC50 = 50 nM T59328 C9ZD2E 11626406 IC50 = 1029 nM T59328 CSM62L 11626920 IC50 > 30000 nM T59328 CGX96V 11626927 IC50 < 10000 nM T59328 C1VOW6 11627264 IC50 = 91 nM T59328 CQK9C3 11627337 IC50 < 1 nM T59328 C65ZXO 11632139 IC50 = 10000 nM T59328 CG0K4A 11632391 IC50 = 1.7 nM T59328 CK34LS 11632737 IC50 > 50000 nM T59328 CR1GI3 11633096 IC50 = 9 nM T59328 CB4YR6 11634425 IC50 = 17 nM T59328 C19LFT 11634645 IC50 = 5 nM T59328 CFM2Y4 11640405 IC50 > 10000 nM T59328 C3DIA4 11640601 IC50 > 100000 nM T59328 CW5A2S 11640889 IC50 = 32 nM T59328 C9T6SC 11640926 Ki > 1800 nM T59328 CE5MY2 11645981 IC50 = 10000 nM T59328 C9SPF4 11654839 IC50 = 340 nM T59328 C63JRY 11655241 IC50 = 1200 nM T59328 CA8X1L 11655791 IC50 = 0.64 nM T59328 C1AX2K 11656050 IC50 = 12 nM T59328 C79EDK 11657332 IC50 = 15 nM T59328 COI6C7 11660896 IC50 = 0.38 nM T59328 C24GRQ 11661959 IC50 = 20 nM T59328 C59AXH 11663284 IC50 = 16 nM T59328 CP04JC 11666231 IC50 > 10000 nM T59328 C8BLT1 11667173 IC50 = 32.2 nM T59328 CK64UO 11668874 IC50 = 2900 nM T59328 C1ZAE8 11669455 IC50 = 30 nM T59328 C5QM4L 11670167 IC50 = 1430 nM T59328 C9YK5E 11675213 IC50 = 22 nM T59328 CVLA25 11675714 IC50 = 500 nM T59328 CDA46H 11675978 IC50 = 16 nM T59328 C75CNZ 11678194 IC50 = 6.7 nM T59328 C0YOG3 11681189 IC50 = 199.53 nM T59328 C7T9ES 11681588 IC50 = 150 nM T59328 CS72ED 11682843 IC50 = 20 nM T59328 CQ69CR 11683171 IC50 = 204 nM T59328 C9YA5W 11683816 IC50 = 47 nM T59328 CJ9KN7 11683817 IC50 > 10000 nM T59328 C6GQ3R 11684059 IC50 = 1600 nM T59328 CQA9W7 11684098 IC50 = 150 nM T59328 C1P8JC 11684684 IC50 = 7 nM T59328 CP3U0W 11684933 IC50 = 397 nM T59328 C8AEX7 11687971 IC50 > 200000 nM T59328 C0UGQ3 11689490 IC50 = 10000 nM T59328 CU0E8O 11690457 Ki > 10000 nM T59328 C5JNW3 11690494 IC50 > 100000 nM T59328 C7I9FP 11690513 IC50 = 700 nM T59328 CLC53E 11691173 IC50 = 10 nM T59328 CP8WJ3 11691483 IC50 > 10000 nM T59328 C6QI9A 11698674 IC50 = 38 nM T59328 CKF8X5 11698913 IC50 = 13 nM T59328 C5J8NA 11703562 IC50 = 17 nM T59328 CX6IC8 11705545 IC50 > 100000 nM T59328 CB0AP2 11705863 Ki > 10000 nM T59328 CI7O1T 11706282 IC50 = 97 nM T59328 C1XNT2 11710303 IC50 = 99 nM T59328 CXOF82 11711590 IC50 = 15 nM T59328 CLY3T0 11712237 IC50 = 1100 nM T59328 CWX07A 11712609 IC50 = 216 nM T59328 C93EKF 11712721 IC50 = 70 nM T59328 CXKT32 11712931 IC50 = 1.66 nM T59328 C4YWU2 11713043 IC50 = 4.5 nM T59328 CR51YI 11717370 IC50 = 676 nM T59328 C1FTX3 11719305 IC50 = 35 nM T59328 CZY05V 11719421 IC50 = 965 nM T59328 C8WQ9F 11719423 IC50 = 4.2 nM T59328 CC3XP1 11720499 IC50 = 23 nM T59328 C8QI0K 11723086 IC50 > 20000 nM T59328 CFJ4I7 11723151 IC50 > 100000 nM T59328 C45EWD 11723489 IC50 > 7000 nM T59328 C9HC4M 11726643 IC50 = 3900 nM T59328 C9P0VD 11729539 IC50 > 100000 nM T59328 CQ3R5E 11733863 IC50 = 130 nM T59328 C7C2FM 11737638 IC50 > 100000 nM T59328 CPY1Z2 11740563 IC50 = 800 nM T59328 CP7AH3 11755812 IC50 = 50000 nM T59328 CWL34S 11756855 IC50 > 100000 nM T59328 C43NTX 11762902 IC50 = 550 nM T59328 C3J7MT 11777791 IC50 > 100000 nM T59328 CGYV23 11779501 IC50 = 360 nM T59328 C9Z7WU 11779874 IC50 > 20000 nM T59328 CV2RD0 11786660 IC50 = 140 nM T59328 CTZ60E 11786930 IC50 = 32 nM T59328 CF2M6O 11797642 IC50 > 20000 nM T59328 CJPT37 11799155 IC50 = 1.5 nM T59328 CH37DA 11802348 IC50 = 3000 nM T59328 C4Q1AE 11817879 IC50 = 110 nM T59328 CYO7K5 11822927 IC50 = 482 nM T59328 C9JT4S 11847343 IC50 > 10000 nM T59328 CHR92S 11858109 IC50 = 1700 nM T59328 CQF23E 11952856 IC50 < 10 nM T59328 C0A4TX 11955109 IC50 = 3 nM T59328 CESM43 11955112 IC50 = 9 nM T59328 CAGY67 11955434 IC50 = 13 nM T59328 CM50UH 12000646 IC50 > 10000 nM T59328 CKPW61 12211388 IC50 = 2710 nM T59328 C2Y5BU 12213273 IC50 = 10 nM T59328 CD6KA7 12241082 IC50 = 2 ug.mL-1 T59328 CJ5K4M 12341776 IC50 = 52 nM T59328 C78FCI 12482705 IC50 = 20040 nM T59328 C9MHX7 12484326 IC50 > 100000 nM T59328 C6PYI9 12814948 IC50 = 75000 nM T59328 C40ZMY 13038269 IC50 = 156 nM T59328 C0NBY4 13041145 IC50 = 1080 nM T59328 CT0R3M 13126887 IC50 = 30 nM T59328 CWUK08 13492269 IC50 = 1900 nM T59328 CO74KJ 13492270 IC50 = 2100 nM T59328 C9J0ID 13492273 IC50 = 77500 nM T59328 CHD0C6 13492275 IC50 = 75100 nM T59328 CR1H5O 13492276 IC50 > 50000 nM T59328 C7LN2W 13492279 IC50 = 560 nM T59328 CJXA95 13492280 IC50 = 1900 nM T59328 C2QEX8 13492281 IC50 = 3000 nM T59328 CC16HJ 13492282 IC50 = 110 nM T59328 CE0IS9 13492283 IC50 > 100000 nM T59328 CC70UD 13498036 IC50 > 100000 nM T59328 CG0VW8 13965155 IC50 = 17190 nM T59328 C5MI4N 14246200 IC50 = 60 nM T59328 CXPU45 14246203 IC50 = 110 nM T59328 C52VQJ 14459363 IC50 = 20 ug.mL-1 T59328 CY1I9N 14459364 IC50 = 2 ug.mL-1 T59328 C2HK6N 14459365 IC50 = 5 ug.mL-1 T59328 CRB23M 14489592 IC50 = 412.3 nM T59328 CQA20E 14547432 IC50 = 20000 nM T59328 C2Z8DQ 14624081 IC50 = 4600 nM T59328 C05MWB 14738184 IC50 = 31768.74 nM T59328 CY6H5R 14758720 IC50 = 56.48 nM T59328 CQ2MO7 14800296 IC50 > 6 ug.mL-1 T59328 CJ1XI6 14800297 IC50 > 6 ug.mL-1 T59328 CCG0R9 14862523 IC50 = 2800 nM T59328 C9EOJ3 14862524 IC50 = 50 nM T59328 CZ4C8O 14862525 IC50 = 300 nM T59328 C8ID0S 14862526 IC50 = 2500 nM T59328 C8AF0C 14862527 IC50 = 1500 nM T59328 CMIY48 14862528 IC50 = 1800 nM T59328 CLQJ06 14862530 IC50 = 600 nM T59328 CO1WA7 14862532 IC50 = 500 nM T59328 C4P3OG 14862533 IC50 = 400 nM T59328 CICQ96 14862534 IC50 = 4000 nM T59328 C3HEO0 14862536 IC50 = 1300 nM T59328 CAJ79W 14862537 IC50 = 4800 nM T59328 CAY7Z2 14862538 IC50 > 100000 nM T59328 CI5KD3 14862539 IC50 = 1000 nM T59328 CTM1N7 14862540 IC50 = 5000 nM T59328 CK60ZN 14862550 IC50 > 50000 nM T59328 CHC25I 14862551 IC50 = 20000 nM T59328 CUMI23 14943555 IC50 = 15000 nM T59328 CRZG26 14943556 IC50 = 6100 nM T59328 C5M6ZT 14943557 IC50 = 28700 nM T59328 CJ5RZ6 14994201 IC50 = 400 nM T59328 CW48TD 15159374 IC50 = 689 nM T59328 CK8XF4 15209376 IC50 = 1500 nM T59328 CPK05U 15249955 IC50 = 100000 nM T59328 CDGF78 15282555 IC50 = 1300 nM T59328 CVU54Q 15324448 IC50 = 19730 nM T59328 CIL1R3 15411595 IC50 = 160000 nM T59328 CKU75C 15520888 IC50 = 1643.6 nM T59328 CQ9Z0L 15550318 IC50 = 5100 nM T59328 CW4R6I 15550657 IC50 = 374.8 nM T59328 CJ81ZO 15550658 IC50 = 6266.2 nM T59328 CN2Z1V 15598735 IC50 = 10 ug.mL-1 T59328 CL81NH 15598736 IC50 = 10 ug.mL-1 T59328 C01JGR 15598739 IC50 = 5 ug.mL-1 T59328 CR7SM0 15598740 IC50 = 4 ug.mL-1 T59328 CSFP09 15598743 IC50 = 2 ug.mL-1 T59328 CAG6P9 15598744 IC50 = 10 ug.mL-1 T59328 C6JS5O 15603105 IC50 = 5.35 nM T59328 CP8OW6 15858662 IC50 = 500 nM T59328 CUI6E5 15858664 IC50 = 170 nM T59328 C6PZU3 15858665 IC50 = 350 nM T59328 CEMH32 15858666 IC50 = 1530 nM T59328 CK5QI3 15858667 IC50 = 1120 nM T59328 CFHW20 15942947 IC50 = 85600 nM T59328 C1O8MK 15946672 IC50 = 9 nM T59328 C7LB4I 15949613 IC50 > 10000 nM T59328 C21YPU 16004616 IC50 = 90400 nM T59328 CFPW41 16007116 Ki > 1800 nM T59328 CS28LD 16035342 IC50 = 40 nM T59328 C5KS0Q 16036986 IC50 = 10 nM T59328 CQM4R7 16036987 IC50 = 15 nM T59328 CBU5P8 16037083 IC50 = 12 nM T59328 C69NIP 16037084 IC50 = 13 nM T59328 CM8IN2 16037085 IC50 = 4 nM T59328 C91PSH 16037086 IC50 = 12 nM T59328 CDZR21 16037089 IC50 = 25 nM T59328 CZ0UJ7 16037184 IC50 = 43 nM T59328 CAZ34B 16037276 IC50 = 3300 nM T59328 C1DO0X 16037278 IC50 = 187 nM T59328 CQR5O7 16042971 IC50 = 1500 nM T59328 CZK8V6 16043304 IC50 > 10000 nM T59328 CH9LO8 16044634 IC50 = 7700 nM T59328 C3ZC6E 16045442 IC50 < 1 nM T59328 C2MH6N 16045730 IC50 = 1 nM T59328 CD2F8V 16046116 IC50 = 690 nM T59328 CQW10N 16066845 IC50 = 30 nM T59328 C3GW0S 16069809 IC50 = 83900 nM T59328 CQG45C 16109001 IC50 = 25000 nM T59328 CZC0H1 16116961 IC50 = 180 nM T59328 C6D8MB 16118310 Ki = 1.6 nM T59328 CL5IF2 16214946 IC50 > 30000 nM T59328 CY1CB3 16215851 IC50 = 60 nM T59328 CXUO14 16457485 IC50 = 311 nM T59328 CVCD64 16663769 IC50 = 0.1 nM T59328 CU56EW 16664858 IC50 > 10000 nM T59328 C2IF3P 16678352 IC50 = 3580 nM T59328 C3IO1C 16679060 IC50 > 10000 nM T59328 C5WIS9 16719846 IC50 = 71 nM T59328 CCD20J 16719847 IC50 = 2200 nM T59328 CT68JW 16719965 IC50 = 970 nM T59328 C02KXR 16719966 IC50 = 4.4 nM T59328 CMLX63 16719967 IC50 = 3960 nM T59328 CHZ20P 16730263 IC50 = 20 nM T59328 C1Y2JH 16745310 IC50 = 799.3 nM T59328 CN8WX3 16757526 IC50 = 22000 nM T59328 CEXL56 17271861 IC50 = 13230 nM T59328 CQY57T 17747104 IC50 = 70 nM T59328 C4BQ6L 17747105 IC50 = 8 nM T59328 CKU29X 17747134 IC50 = 12 nM T59328 C5YZ9V 17747138 IC50 = 16 nM T59328 C95LWR 17747139 IC50 = 5 nM T59328 CW61OK 17747208 IC50 = 32 nM T59328 CQ7RH3 17747242 IC50 = 13 nM T59328 CXD23O 17747243 IC50 = 24 nM T59328 C2VL8S 17747279 IC50 = 47 nM T59328 C8AM0W 17747280 IC50 = 23 nM T59328 CEG7O8 17747281 IC50 = 14 nM T59328 CR4PF2 17747282 IC50 = 44 nM T59328 CYB3N5 17747309 IC50 = 20 nM T59328 CC2W0F 17747311 IC50 = 23 nM T59328 CS9O2H 17747339 IC50 = 48 nM T59328 CL83TA 17747341 IC50 = 104 nM T59328 C1VC9E 17747343 IC50 = 14 nM T59328 C7Q0ZD 17747376 IC50 = 57 nM T59328 CUT1G2 17747492 IC50 = 33 nM T59328 CNRV46 17747535 IC50 = 27 nM T59328 CL9BQ6 17748275 IC50 = 25000 nM T59328 CAV9R6 17757434 IC50 > 20000 nM T59328 C8AH1I 17758019 IC50 = 1000 nM T59328 C1GKL6 17758020 IC50 > 5000 nM T59328 CO6LR5 17758240 IC50 = 500 nM T59328 CU0MF7 17758241 IC50 = 3300 nM T59328 CE73IF 17758353 IC50 = 5000 nM T59328 CH9TR6 17758354 IC50 = 156 nM T59328 CA79FH 17758358 IC50 > 5000 nM T59328 CSA23C 17759556 IC50 > 20000 nM T59328 C56YOG 17759673 IC50 = 2080 nM T59328 CIL8G9 17759675 IC50 > 20000 nM T59328 C57NRL 17759787 IC50 = 2900 nM T59328 C3D7WE 17874201 IC50 > 200000 nM T59328 C35IWY 17938625 IC50 = 4000 nM T59328 C7ZK1E 17938633 IC50 = 30000 nM T59328 CQ35AK 17953498 IC50 = 730 nM T59328 CM2HS9 18176200 IC50 = 0.6 nM T59328 C60VEN 18176234 IC50 = 0.69 nM T59328 CYD95N 18184369 IC50 = 132 nM T59328 C8NCX0 18184376 IC50 = 2110 nM T59328 C1SQC4 18184420 IC50 = 72 nM T59328 CQA78V 18382736 IC50 = 5 nM T59328 C2EBQ5 18382775 IC50 = 4 nM T59328 CZB5L4 18382784 IC50 = 100 nM T59328 C1LUP2 18382794 IC50 = 3 nM T59328 C8KJ4R 18382823 IC50 > 1000 nM T59328 CZC98J 18382853 IC50 = 1 nM T59328 C5QV1L 18382857 IC50 = 1600 nM T59328 C84KLY 18382861 IC50 = 30 nM T59328 CSPD61 18382868 IC50 = 140 nM T59328 CG4BK9 18382875 IC50 = 3 nM T59328 C8BK3Q 18382898 IC50 = 4 nM T59328 CX7F1I 18382902 IC50 = 2 nM T59328 CNE4R0 18382910 IC50 = 1 nM T59328 CML03B 18382946 IC50 = 5 nM T59328 CGXU47 18382956 IC50 = 600 nM T59328 C5BGJ8 18382993 IC50 = 2 nM T59328 CVFU60 18383007 IC50 = 9 nM T59328 CZ90LJ 18383038 IC50 = 9 nM T59328 C2R0KU 18383095 IC50 = 94 nM T59328 CBF6H0 18383099 IC50 = 500 nM T59328 C7SQ3Z 18383101 IC50 = 657 nM T59328 CQ7V2F 18383102 IC50 = 250 nM T59328 CT7GK6 18548938 IC50 > 10000 nM T59328 CX69ZL 18548951 IC50 > 10000 nM T59328 C8MQ2N 18770775 IC50 = 5500 nM T59328 CY97MC 18770784 IC50 = 100 nM T59328 CHDY96 18770788 IC50 = 600 nM T59328 C1HCE3 18770799 IC50 = 3000 nM T59328 C72EWO 18770811 IC50 = 6500 nM T59328 C4BTV7 18770818 IC50 = 3000 nM T59328 C3JP7K 18770822 IC50 > 20000 nM T59328 C1GAJ2 18770840 IC50 = 500 nM T59328 C1C0EJ 18792861 IC50 = 2540 nM T59328 C6HK0S 18792868 IC50 = 500 nM T59328 C90EQY 18792940 IC50 = 2670 nM T59328 C9PS7R 18792941 IC50 = 900 nM T59328 CIH2K0 18792942 IC50 = 400 nM T59328 CILQ48 18792962 IC50 = 13400 nM T59328 C7R5VZ 18967573 IC50 = 59 nM T59328 C3AZJ2 19037238 IC50 > 200000 nM T59328 CC7U2Q 19077486 IC50 = 79 nM T59328 CXB56W 19077488 IC50 = 57 nM T59328 C96VSF 19077498 IC50 = 49 nM T59328 CNC8P2 19077501 IC50 = 7 nM T59328 C54VNA 19077504 IC50 = 61 nM T59328 C3O9AD 19077506 IC50 = 60.2 nM T59328 CEO7V9 19077507 IC50 = 98 nM T59328 CAUO09 19077508 IC50 = 10 nM T59328 CMI72S 19077513 IC50 = 93 nM T59328 CU4R5O 19077515 IC50 = 18.1 nM T59328 CB32XU 19077516 IC50 = 71 nM T59328 CBUP69 19077520 IC50 = 87 nM T59328 C0FL3G 19888887 IC50 > 30 ug.mL-1 T59328 C0WEX3 19966997 IC50 > 100000 nM T59328 C0E2OG 20579089 IC50 > 10000 nM T59328 C3AI0N 20817111 IC50 = 2300 nM T59328 CFI0B9 21010047 IC50 = 2.61 nM T59328 C81ALS 21080010 IC50 = 0.11 nM T59328 C51HNQ 21080015 IC50 = 0.94 nM T59328 CL81VC 21100709 IC50 = 100000 nM T59328 C3EHM4 21197160 IC50 = 90000 nM T59328 CEBF05 21697320 IC50 = 150 nM T59328 CVI49J 21701562 IC50 = 5700 nM T59328 CFN6G4 21701597 IC50 = 100 nM T59328 C5B7WP 21874200 IC50 = 9 nM T59328 CBN19I 21874228 IC50 = 130 nM T59328 CLD73T 21874248 IC50 = 32 nM T59328 CYSR48 21874287 IC50 = 20 nM T59328 CWY6T7 21874402 IC50 = 660 nM T59328 C5IBJ0 21874410 IC50 = 6 nM T59328 CM3XF9 21874431 IC50 = 50 nM T59328 CRB1V5 21945809 IC50 = 490 nM T59328 CT9LP3 21945841 IC50 = 200 nM T59328 C5GIE9 21945968 IC50 = 40 nM T59328 CHU2Z3 21951965 IC50 = 80 nM T59328 CLN2G9 21952043 IC50 = 25 nM T59328 CH27DF 21988185 IC50 > 10000 nM T59328 COH4Y2 21988214 IC50 > 10000 nM T59328 CXJI39 22022153 IC50 = 100 nM T59328 CFG57O 22024915 IC50 = 2 nM T59328 C5MEX2 22024916 IC50 = 150 nM T59328 CQEN87 22055240 IC50 = 85 nM T59328 C8J9GH 22055262 IC50 = 48 nM T59328 C2RY4D 22055269 IC50 = 250 nM T59328 CPV5Z0 22132688 IC50 > 10000 nM T59328 CH5V2Q 22390479 IC50 = 210 nM T59328 C1IU0K 22390480 IC50 = 710 nM T59328 C50SLD 22390490 IC50 = 620 nM T59328 C7GK1A 22390495 IC50 = 110 nM T59328 CKV0J5 22390502 IC50 = 500 nM T59328 C5NVM0 22390522 IC50 = 220 nM T59328 C9G5RQ 22390524 IC50 = 50 nM T59328 CHF3A0 22390530 IC50 = 100 nM T59328 CD5GI0 22390536 IC50 = 110 nM T59328 C18CUK 22390541 IC50 = 200 nM T59328 C3H4NO 22390542 IC50 = 120 nM T59328 CNMZ85 22390556 IC50 = 380 nM T59328 C1CJS9 22466664 IC50 = 330.2 nM T59328 CWL0O9 22466767 IC50 = 1040 nM T59328 CF6LA9 22478260 IC50 = 90 nM T59328 CMRO51 22478297 IC50 = 80 nM T59328 C7TK3G 22478429 IC50 = 126.9 nM T59328 C2P1DL 22667101 IC50 > 10000 nM T59328 CK35BP 22667145 IC50 > 10000 nM T59328 C1PR6W 22692676 IC50 > 50000 nM T59328 CSB1G3 22692751 IC50 = 900 nM T59328 CYN49O 22692759 IC50 = 37600 nM T59328 CZRM03 22692773 IC50 = 36000 nM T59328 CB1V6E 22692848 IC50 = 2370 nM T59328 CO2R3S 22692946 IC50 = 4300 nM T59328 C9WHT0 22692968 IC50 > 100000 nM T59328 CKB7C2 22693031 IC50 > 100000 nM T59328 C6CHV3 22693234 IC50 = 9700 nM T59328 CC1U4X 22732253 IC50 = 5600 nM T59328 COB60M 23133320 IC50 = 100 nM T59328 C9QLP0 23133323 IC50 = 170 nM T59328 C4E1SO 23290441 IC50 = 0.208 nM T59328 CQMH63 23366746 IC50 = 1800 nM T59328 C6JV7W 23400934 IC50 > 7000 nM T59328 CD5S7O 23401001 IC50 > 7000 nM T59328 CV8P7G 23546054 IC50 > 40000 nM T59328 C9PF3L 23546055 IC50 = 5400 nM T59328 C2XRV0 23546056 IC50 = 1000 nM T59328 CWU9P6 23589545 IC50 = 120 nM T59328 CEN3B8 23589555 IC50 = 950 nM T59328 CRX0Q6 23625758 IC50 > 100000 nM T59328 C19TLD 23644675 IC50 = 1600 nM T59328 CX32IF 23646535 IC50 = 90 nM T59328 C4Z5YE 23646536 IC50 = 60 nM T59328 CZ6E5P 23646537 IC50 = 50 nM T59328 CG7F1M 23646539 IC50 = 610 nM T59328 C9ZSO0 23646540 IC50 = 120 nM T59328 C06CVI 23646541 IC50 = 200 nM T59328 C42ONU 23646542 IC50 = 200 nM T59328 C3T8FB 23646543 IC50 > 25000 nM T59328 CVK4Z2 23646544 IC50 = 120 nM T59328 CS31HG 23646545 IC50 = 70 nM T59328 CRQK51 23646546 IC50 = 210 nM T59328 C7O2QA 23646547 IC50 = 7400 nM T59328 C82MEJ 23646548 IC50 = 950 nM T59328 C08NIK 23646549 IC50 = 1100 nM T59328 CV75ZR 23646550 IC50 = 170 nM T59328 C2S5ZM 23661662 Ki = 3 nM T59328 CYWG82 23729145 IC50 = 490 nM T59328 COV2N4 24179332 IC50 = 10340 nM T59328 CUGY24 24202429 IC50 = 1900 nM T59328 CNWM52 24322804 IC50 = 7440 nM T59328 CLIV79 24737855 IC50 < 15 nM T59328 CH53CN 24738004 IC50 = 5.06 nM T59328 CA3I4T 24753787 IC50 > 50000 nM T59328 C7YG1N 24759534 IC50 = 1100 nM T59328 CAJ4T2 24762205 IC50 > 10000 nM T59328 CCPS81 24764502 IC50 > 35000 nM T59328 C78RNQ 24766872 IC50 = 197 ug.mL-1 T59328 CQ8SY7 24766873 IC50 > 200 ug.mL-1 T59328 C31EHS 24767187 IC50 > 20000 nM T59328 CJUK39 24770517 IC50 > 10000 nM T59328 C0EKO5 24772654 IC50 = 3300 nM T59328 CC1L8F 24777233 IC50 = 76 nM T59328 CXS1U4 24779710 IC50 = 14.1 nM T59328 C1CGU3 24782374 IC50 = 5000 nM T59328 C7DR5J 24782621 IC50 = 257 nM T59328 CFN39G 24782622 IC50 = 980 nM T59328 CE2Q3V 24786207 IC50 = 1160 nM T59328 C9PA0M 24807809 IC50 > 10000 nM T59328 CY8X0J 24811794 Ki > 10000 nM T59328 C7UPH2 24824775 IC50 = 4720 nM T59328 C61KPI 24856363 IC50 > 25000 nM T59328 C3S5KC 24863865 IC50 = 209 nM T59328 CFK2B9 24882503 IC50 = 380 nM T59328 C43HWQ 24883287 IC50 = 24 nM T59328 C8DA5Q 24883334 IC50 = 9 nM T59328 C4V9GH 24894117 IC50 = 23000 nM T59328 CZ6KD4 24894886 IC50 = 22000 nM T59328 CB5TP8 24894992 IC50 = 9000 nM T59328 C32SUJ 24894993 IC50 = 14000 nM T59328 CY8L7E 24896769 IC50 > 10000 nM T59328 CZ67RA 24897043 IC50 = 8 nM T59328 CVF5W2 24897276 IC50 = 30 nM T59328 CB2EX1 24897277 IC50 = 16 nM T59328 CN9T1Z 24897278 IC50 = 16 nM T59328 C6JA7L 24897279 IC50 = 31 nM T59328 CA5XT2 24897280 IC50 = 26 nM T59328 CN13JF 24899915 IC50 = 4.2 ug.mL-1 T59328 CBWR97 24899916 IC50 = 1.1 ug.mL-1 T59328 C9F2JD 24899917 IC50 > 10 ug.mL-1 T59328 C64MTI 24900160 IC50 = 4.2 ug.mL-1 T59328 CO2I6Q 24900161 IC50 = 6.5 ug.mL-1 T59328 CB79YC 24905143 IC50 = 954 nM T59328 C2DC9J 24905144 IC50 = 388 nM T59328 CN6V8Z 24905145 IC50 = 550 nM T59328 CSB7P5 24905148 IC50 = 12000 nM T59328 CGSF21 24905149 IC50 > 50000 nM T59328 CVDG02 24905150 IC50 = 170 nM T59328 CWH6C5 24905152 IC50 = 610 nM T59328 C0HE2Q 24905153 IC50 = 2300 nM T59328 C7QSC9 24905154 IC50 = 579 nM T59328 CO9D0K 24905155 IC50 = 12000 nM T59328 C5W9UR 24905157 IC50 = 9900 nM T59328 CC1DA3 24905158 IC50 = 5960 nM T59328 COW79F 24905159 IC50 = 100000 nM T59328 CFPA53 24905160 IC50 = 100000 nM T59328 C2O0JX 24905161 IC50 = 12800 nM T59328 CA72BE 24905162 IC50 = 100000 nM T59328 CQN6X9 24905163 IC50 = 100000 nM T59328 CD4O1F 24905165 IC50 = 8300 nM T59328 CKL48T 24905166 IC50 = 13000 nM T59328 C76VYL 24905167 IC50 = 17000 nM T59328 C7K5PU 24905168 IC50 = 4300 nM T59328 CZ57ID 24905169 IC50 = 1400 nM T59328 C2DHX9 24905170 IC50 = 100000 nM T59328 CSB96E 24905171 IC50 = 100000 nM T59328 CWZ0R2 24905172 IC50 = 15000 nM T59328 CY3B6M 24905175 IC50 = 3860 nM T59328 CW7UA3 24905176 IC50 = 10200 nM T59328 CW1V0H 24905177 IC50 = 5140 nM T59328 CO6Y0L 24905178 IC50 = 3660 nM T59328 C60NQW 24905179 IC50 = 100000 nM T59328 C4MO8B 24905180 IC50 = 3720 nM T59328 COJI47 24905181 IC50 = 1770 nM T59328 CS0B2C 24905182 IC50 = 751 nM T59328 C1H4BT 24905183 IC50 = 84 nM T59328 C4WHK9 24905184 IC50 = 11000 nM T59328 C7Q4MZ 24905185 IC50 = 179 nM T59328 CS4IP1 24905186 IC50 = 249 nM T59328 C69QWO 24905187 IC50 = 391 nM T59328 C85ANB 24905188 IC50 = 176 nM T59328 CNHD75 24905189 IC50 = 3300 nM T59328 C9JUO2 24905190 IC50 = 4600 nM T59328 CPR03K 24905191 IC50 = 1400 nM T59328 CTAG19 24905193 IC50 = 734 nM T59328 C7VJM5 24905194 IC50 = 5000 nM T59328 CEP1L3 24905195 IC50 = 964 nM T59328 CP68ZD 24905196 IC50 = 575 nM T59328 C8Z0RJ 24905197 IC50 = 768 nM T59328 CN9RT0 24905198 IC50 = 5320 nM T59328 CHI78P 24905200 IC50 = 1000 nM T59328 CO6PE8 24905201 IC50 = 220 nM T59328 CZ63HS 24905202 IC50 = 380 nM T59328 C2X0FC 24905203 IC50 = 2500 nM T59328 C0WCE3 24905204 IC50 = 34000 nM T59328 CNK50B 24905205 IC50 = 2100 nM T59328 C12DPB 24905206 IC50 = 760 nM T59328 C8N0RH 24905207 IC50 = 21000 nM T59328 CYA5G2 24905208 IC50 = 100000 nM T59328 CDV2B4 24905209 IC50 = 2900 nM T59328 CEFK68 24905210 IC50 = 15000 nM T59328 CUFP12 24905211 IC50 = 540 nM T59328 C0JG8L 24905212 IC50 = 85 nM T59328 CQ13ZI 24905215 IC50 = 25000 nM T59328 C6VI8F 24905216 IC50 = 100000 nM T59328 CXNH25 24905217 IC50 = 100000 nM T59328 C2PN9S 24905218 IC50 = 18000 nM T59328 C9O2AL 24905219 IC50 = 18000 nM T59328 CIT7U8 24905220 IC50 = 100000 nM T59328 CMD26S 24905221 IC50 = 955 nM T59328 C4R8WC 24905222 IC50 = 539 nM T59328 C47SHA 24905223 IC50 = 1100 nM T59328 C1DY2R 24905224 IC50 = 571 nM T59328 CS0XF9 24905225 IC50 = 70000 nM T59328 CG5VX2 24905226 IC50 = 6700 nM T59328 C57QEO 24905227 IC50 = 1400 nM T59328 C7CG5E 24905228 IC50 = 7000 nM T59328 CHP5D1 24905229 IC50 = 29000 nM T59328 CXP09S 24905230 IC50 = 100000 nM T59328 CY7XG1 24905231 IC50 = 100000 nM T59328 C7JFQ2 24905232 IC50 = 12000 nM T59328 C2JM1P 24905233 IC50 = 100000 nM T59328 CC3BF0 24905234 IC50 = 10000 nM T59328 CE57FI 24905235 IC50 = 10000 nM T59328 CUP20O 24905236 IC50 = 100000 nM T59328 CLC6Q2 24905237 IC50 = 8900 nM T59328 C9M1GI 24905238 IC50 = 9000 nM T59328 CVD72F 24905239 IC50 = 207 nM T59328 CK38IZ 24905240 IC50 = 2600 nM T59328 CO2V5E 24905241 IC50 = 937 nM T59328 CZBA19 24905244 IC50 = 1200 nM T59328 CQ8OI1 24905246 IC50 = 45000 nM T59328 CIF2J5 24905251 IC50 = 3850 nM T59328 CPTE58 24905252 IC50 = 2120 nM T59328 CP50RD 24905280 IC50 = 1400 nM T59328 CG13ZM 24905281 IC50 = 33 nM T59328 CF0S6X 24905282 IC50 = 5950 nM T59328 C2Z5DN 24905285 IC50 = 12400 nM T59328 CL6GH8 24905286 IC50 = 100000 nM T59328 CKYO98 24905287 IC50 = 663 nM T59328 CRNQ65 24905288 IC50 = 2190 nM T59328 COD7I5 24905289 IC50 = 1670 nM T59328 C4LP7E 24905290 IC50 = 19000 nM T59328 CE9JC2 24905291 IC50 = 100000 nM T59328 C2GI1R 24905292 IC50 = 100000 nM T59328 CHW8C4 24905293 IC50 = 6450 nM T59328 CQF0H1 24905294 IC50 = 437 nM T59328 CNO7X0 24905295 IC50 = 158 nM T59328 C5WRG7 24905296 IC50 = 1400 nM T59328 CQ1S0U 24905297 IC50 = 5080 nM T59328 C4UES7 24905298 IC50 = 1160 nM T59328 CMS69P 24905299 IC50 = 2720 nM T59328 CC0U5M 24905300 IC50 = 67 nM T59328 CW7X6S 24905301 IC50 = 100000 nM T59328 C97IQV 24905302 IC50 = 318 nM T59328 CSJ47V 24905303 IC50 = 100000 nM T59328 CPN74C 24905304 IC50 = 9380 nM T59328 C5CS3N 24905305 IC50 = 2010 nM T59328 CK4XE9 24905307 IC50 = 100000 nM T59328 CTU6Z3 24905308 IC50 = 100000 nM T59328 C9SQX1 24905309 IC50 = 8700 nM T59328 CM75JP 24905310 IC50 = 15600 nM T59328 C9Q2BJ 24905311 IC50 = 12600 nM T59328 C9VUA1 24905312 IC50 = 12400 nM T59328 CU3RS1 24905313 IC50 = 17000 nM T59328 CYG3H2 24905314 IC50 = 2900 nM T59328 CV5Q7O 24905315 IC50 = 366 nM T59328 C8SA3O 24905316 IC50 = 270 nM T59328 CI5MN3 24905317 IC50 = 1580 nM T59328 CJ1P7K 24905318 IC50 = 1400 nM T59328 C1T6YQ 24905319 IC50 = 4800 nM T59328 CAU86X 24905320 IC50 = 2600 nM T59328 C54ISY 24905321 IC50 = 100000 nM T59328 C2GE5I 24905322 IC50 = 4800 nM T59328 C8D6YK 24905323 IC50 = 26000 nM T59328 C5NZH9 24905324 IC50 = 9140 nM T59328 C9D6JR 24905325 IC50 = 2900 nM T59328 CLZT41 24905326 IC50 = 1150 nM T59328 CW8FD3 24905327 IC50 = 775 nM T59328 CHB7A2 24905328 IC50 = 18000 nM T59328 CA8EI3 24905329 IC50 = 11000 nM T59328 CCQ0O7 24905330 IC50 = 6340 nM T59328 CJ81AS 24905331 IC50 = 100000 nM T59328 C8PW4H 24905332 IC50 = 324 nM T59328 C2Y5TF 24905333 IC50 = 236 nM T59328 CH9FL5 24905334 IC50 = 18000 nM T59328 C1S0PC 24905335 IC50 = 12000 nM T59328 C8N9MV 24905336 IC50 = 4320 nM T59328 C9E8BJ 24905338 IC50 = 100000 nM T59328 CX85AC 24905341 IC50 = 100000 nM T59328 CKZ80E 24905342 IC50 = 576 nM T59328 CO8SH1 24905343 IC50 = 3020 nM T59328 C7IZL6 24905344 IC50 = 100000 nM T59328 C5ZM4T 24936119 IC50 = 2400 nM T59328 C96GPD 24944848 IC50 = 7.1 nM T59328 CNMB03 24944849 IC50 = 7.8 nM T59328 CTCB27 24944850 IC50 = 9.4 nM T59328 C5PH0N 24944851 IC50 = 3.4 nM T59328 CK17HZ 24944855 IC50 = 8.2 nM T59328 C0BOJ2 24944856 IC50 = 7 nM T59328 CX05SV 24944930 IC50 = 3.1 nM T59328 CB8EZ0 24944934 IC50 = 15 nM T59328 C2CP6T 24944935 IC50 = 4.6 nM T59328 C1NZ8X 24945115 IC50 = 84.2 nM T59328 CF0U4T 24945204 IC50 = 10.4 nM T59328 C8W3YA 24945368 IC50 = 2.1 nM T59328 C2MYN7 24945689 IC50 = 9.08 nM T59328 C4V9GI 24960018 IC50 > 20000 nM T59328 C9B7PH 24970496 IC50 = 533 nM T59328 CGV1Q5 24970497 IC50 = 472 nM T59328 C4EG8R 24993189 IC50 > 10000 nM T59328 CHOK82 25000333 IC50 = 42 nM T59328 CBK82P 25011729 IC50 > 30000 nM T59328 CRO0Y8 25022735 IC50 = 122000 nM T59328 C72AJM 25022736 IC50 > 200000 nM T59328 CIK6V8 25025888 IC50 = 3.1 nM T59328 C0JGL8 25026082 IC50 = 3 nM T59328 CHY93R 25026085 IC50 = 8.8 nM T59328 C3DPS2 25026281 IC50 = 1.9 nM T59328 CD8IP2 25039251 IC50 = 12110 nM T59328 CHLQ49 25063262 IC50 = 30 nM T59328 C2KY1G 25094210 IC50 = 5048 nM T59328 C96EVA 25118036 IC50 = 8 nM T59328 CTV54O 25123227 IC50 > 10000 nM T59328 CG3XC9 25124150 IC50 = 57 nM T59328 CO2IR5 25124816 IC50 > 10000 nM T59328 C6BWZ8 25145145 IC50 > 100 nM T59328 C78YWA 25145716 IC50 > 500 nM T59328 CB21XV 25164469 Ki > 1800 nM T59328 CUX83H 25164675 Ki > 1800 nM T59328 C1H7BF 25164677 Ki > 1800 nM T59328 C6SD2A 25165081 Ki > 1800 nM T59328 C67TVH 25165085 Ki > 1800 nM T59328 CRJ6M7 25165279 Ki = 67 nM T59328 C7RBX0 25165280 Ki = 27 nM T59328 CPEY29 25165481 Ki = 17 nM T59328 C70DRX 25165482 Ki = 8 nM T59328 C6VZU2 25165861 Ki > 1800 nM T59328 CGUC69 25167072 Ki > 1800 nM T59328 CF4G1L 25167074 Ki > 1800 nM T59328 C35ZXL 25167075 Ki > 1800 nM T59328 C2D3FP 25167078 Ki > 1800 nM T59328 C37YSX 25167280 Ki > 1800 nM T59328 CX0O5A 25178331 IC50 = 9500 nM T59328 CIG4H0 25178539 IC50 = 4600 nM T59328 C4GI6J 25178540 IC50 = 9900 nM T59328 COB9G8 25181586 IC50 = 15070 nM T59328 CVY98J 25191769 Ki = 18 nM T59328 CP47JK 25192054 Ki = 43 nM T59328 C8K1YN 25192202 Ki = 290 nM T59328 C8TSW4 25192224 IC50 = 290 nM T59328 CBLF93 25192363 IC50 = 50 nM T59328 C09LAT 25192905 Ki = 49 nM T59328 CJ3YN8 25195273 IC50 = 12 nM T59328 C8NBA6 25195274 IC50 = 1 nM T59328 C6FGQ1 25206346 IC50 > 10000 nM T59328 C6XQB9 25207010 IC50 = 44 nM T59328 CRO09K 25211064 IC50 = 10 nM T59328 C8IJB9 25218207 IC50 = 10410 nM T59328 CR0FO4 25218688 EC50 = 335 nM T59328 CWNY70 25218689 EC50 = 742 nM T59328 CZ5M3A 25218690 EC50 = 520 nM T59328 CK9AO6 25218691 EC50 = 808 nM T59328 CXH7F8 25218692 EC50 = 85 nM T59328 CH2GL3 25218693 EC50 = 91 nM T59328 CU49HG 25218695 IC50 = 71 nM T59328 CU0YJ1 25218696 IC50 = 69 nM T59328 CQ6MZ0 25242463 IC50 = 54 nM T59328 CK7ZR2 25242643 IC50 = 320 nM T59328 CM31HJ 25263246 IC50 = 50 nM T59328 CAMY28 25263247 IC50 = 120 nM T59328 C6FB3N 25263248 IC50 = 2600 nM T59328 C7P4FS 25263249 IC50 = 1050 nM T59328 CV8Y5M 25263250 IC50 = 190 nM T59328 CKG21S 25263251 IC50 = 400 nM T59328 C7I4BG 25263252 IC50 = 280 nM T59328 C9TK3Q 25263253 IC50 = 180 nM T59328 CWE9C6 25263254 IC50 = 240 nM T59328 C9SL4P 25263255 IC50 = 1650 nM T59328 C4JQD8 25263256 IC50 = 630 nM T59328 CED02Z 25263257 IC50 = 80 nM T59328 CI79QB 25263258 IC50 = 30 nM T59328 C18VBO 25263259 IC50 = 33 nM T59328 CN89CY 25263260 IC50 = 120 nM T59328 C9JR3E 25263261 IC50 = 230 nM T59328 C0Y9TK 25263263 IC50 = 90 nM T59328 C5I4UQ 25263264 IC50 = 3160 nM T59328 CA0X9R 25263265 IC50 = 680 nM T59328 CW2J5P 25263266 IC50 = 240 nM T59328 CR7JS1 25263267 IC50 = 40 nM T59328 CT60US 25263268 IC50 = 50 nM T59328 C1NAD7 25263269 IC50 = 50 nM T59328 CJI43L 25263270 IC50 = 99 nM T59328 CANP37 25263271 IC50 = 63 nM T59328 CG3OH9 25263272 IC50 = 40 nM T59328 CZ0H9E 25263273 IC50 = 50 nM T59328 CY6HW8 25263274 IC50 = 40 nM T59328 C1WG7S 25263275 IC50 = 40 nM T59328 C6WV8D 25263276 IC50 = 125 nM T59328 CJW7I3 25263277 IC50 = 79 nM T59328 CTO10V 25263278 IC50 = 79 nM T59328 CZ4HN9 25263279 IC50 = 32 nM T59328 C7XEB3 25263280 IC50 = 79 nM T59328 C2ICK6 25263281 IC50 = 50 nM T59328 CZGQ83 25271178 IC50 = 41 nM T59328 CF2LZ7 25271179 IC50 = 150 nM T59328 CUAK50 25271517 IC50 = 76 nM T59328 CU09IM 26699441 IC50 = 50000 nM T59328 C69PNL 40433957 IC50 = 48600 nM T59328 CVM13K 42596931 IC50 = 42 nM T59328 CU53WB 42596953 IC50 = 18 nM T59328 CG2IJ8 42601891 IC50 < 1 nM T59328 C41TLH 42603880 IC50 = 35000 nM T59328 CS1AT2 42603881 IC50 = 93000 nM T59328 CZ2VH7 42604008 IC50 = 82000 nM T59328 CV1P3W 42604009 IC50 = 89000 nM T59328 CWS37O 42618140 IC50 > 10000 nM T59328 C2JV3O 42618143 IC50 > 10000 nM T59328 CG01BO 42618144 IC50 > 10000 nM T59328 CU9E4P 42629114 IC50 > 10000 nM T59328 CR5XJ4 42630202 IC50 = 7130 nM T59328 CJ5U1X 42639664 IC50 = 2.7 ug.mL-1 T59328 CPS5F6 43517028 IC50 = 6.2 nM T59328 CO42DC 44138048 IC50 > 10000 nM T59328 CL65QV 44138049 IC50 > 10000 nM T59328 CUX7D9 44143345 IC50 = 1000 nM T59328 C8YN5P 44143370 IC50 = 11000 nM T59328 C9CWO1 44143371 IC50 = 30000 nM T59328 C26XFL 44143372 IC50 = 22000 nM T59328 C5SEQ2 44143373 IC50 = 22000 nM T59328 CTN41Y 44156909 IC50 = 240 nM T59328 CN0X1C 44156917 IC50 = 63 nM T59328 CB0O2A 44186880 Ki > 1800 nM T59328 C9K7OP 44186882 Ki > 1800 nM T59328 CX0ZU8 44186885 Ki > 1800 nM T59328 CCFQ29 44187005 IC50 = 173 nM T59328 CNGV37 44189584 Ki > 1800 nM T59328 C2AV1K 44190762 IC50 = 2240 nM T59328 C6U2LF 44205208 IC50 = 4.1 nM T59328 CR03OF 44229775 IC50 = 2.9 nM T59328 CEL61X 44229839 IC50 = 2.6 nM T59328 C8DWO1 44229840 IC50 = 7 nM T59328 CNM3H2 44229841 IC50 = 21 nM T59328 C4NWP5 44246325 IC50 = 2200 nM T59328 C2EW0I 44246326 IC50 = 18200 nM T59328 CSD8T0 44246327 IC50 = 56500 nM T59328 CMKF08 44246328 IC50 = 13400 nM T59328 CAO87V 44246329 IC50 > 500000 nM T59328 CLU2V3 44246330 IC50 > 200000 nM T59328 CHZ6Q1 44269004 IC50 > 20000 nM T59328 C83QHW 44273476 IC50 > 100000 nM T59328 C8PT0I 44273491 IC50 > 200000 nM T59328 CS6NT3 44273526 IC50 = 100000 nM T59328 CG8H3R 44273527 IC50 > 200000 nM T59328 C7I1NX 44273528 IC50 = 95000 nM T59328 C3EFQ0 44273554 IC50 > 100000 nM T59328 CAJ48G 44273555 IC50 > 100000 nM T59328 C6VYU1 44273559 IC50 = 49000 nM T59328 C1WAE7 44273560 IC50 > 200000 nM T59328 CQEW06 44273561 IC50 > 200000 nM T59328 C82YSI 44273595 IC50 > 100000 nM T59328 CUG08T 44273597 IC50 > 200000 nM T59328 CIC13W 44273598 IC50 > 200000 nM T59328 CC8W2J 44273599 IC50 > 200000 nM T59328 CR1M9A 44273600 IC50 = 59000 nM T59328 CE6F2M 44273605 IC50 > 200000 nM T59328 CBV2Y3 44273617 IC50 > 200000 nM T59328 CAK08Y 44273618 IC50 = 90000 nM T59328 C0HG8U 44273619 IC50 = 75000 nM T59328 CMRX16 44273620 IC50 > 100000 nM T59328 CT79EW 44273623 IC50 > 200000 nM T59328 CZ6SM5 44273624 IC50 > 200000 nM T59328 CA8J9D 44273646 IC50 > 200000 nM T59328 C8JWQ2 44273647 IC50 = 180000 nM T59328 CI72SY 44273652 IC50 > 200000 nM T59328 CB0IL4 44273653 IC50 > 200000 nM T59328 CA6LH1 44273654 IC50 > 200000 nM T59328 C35TZW 44273659 IC50 > 100000 nM T59328 C8U2RI 44273699 IC50 > 200000 nM T59328 CY9LQ3 44273700 IC50 > 200000 nM T59328 CS7V9G 44278848 IC50 = 1.7 nM T59328 CIYC41 44279645 IC50 = 3762.4 nM T59328 CYEW69 44279647 IC50 = 2043.6 nM T59328 CMU95A 44285249 IC50 = 8.8 nM T59328 CO80RB 44285309 IC50 > 10000 nM T59328 CJQD03 44286273 IC50 = 350 nM T59328 CW02AS 44294903 IC50 > 50000 nM T59328 CRV54Q 44297168 IC50 = 11 nM T59328 C0RIG2 44297343 IC50 = 7 nM T59328 C5N7TD 44297358 IC50 = 120 nM T59328 C8ZAC4 44297408 IC50 = 4 nM T59328 CW0QU5 44299755 IC50 = 69 nM T59328 C2UZ3J 44299923 IC50 = 5 nM T59328 CT72NU 44299926 IC50 = 6 nM T59328 CD91OZ 44299938 IC50 = 5 nM T59328 CE2IC7 44299956 IC50 = 8 nM T59328 C72APV 44299983 IC50 = 8 nM T59328 C5ZSM3 44300005 IC50 = 2 nM T59328 C6CK9A 44300029 IC50 = 310 nM T59328 CFIO61 44300050 IC50 = 100 nM T59328 CJ7A3Y 44300081 IC50 = 8 nM T59328 CO25AL 44300251 IC50 = 35 nM T59328 CW6J2V 44313484 IC50 > 50000 nM T59328 C30GOH 44315116 IC50 = 17000 nM T59328 CA3C4I 44315117 IC50 > 50000 nM T59328 CMN04X 44315118 IC50 = 7000 nM T59328 CS8WZ6 44315309 IC50 = 40000 nM T59328 CUFQ79 44315416 IC50 = 55000 nM T59328 CKD14Y 44316725 IC50 = 1 nM T59328 CM2A1F 44316744 IC50 = 1 nM T59328 CLJ2P3 44316765 IC50 = 1 nM T59328 CK9L3S 44316797 IC50 = 7 nM T59328 C8IAY4 44316957 IC50 = 5 nM T59328 CD69PV 44317138 IC50 = 1 nM T59328 CY6P9K 44318047 IC50 = 70000 nM T59328 CSY8A3 44321301 IC50 = 19000 nM T59328 CCG2M5 44321317 IC50 = 9500 nM T59328 CY9ED1 44321395 IC50 > 100000 nM T59328 C5U1CR 44321686 IC50 > 10000 nM T59328 CETY53 44321717 IC50 > 100000 nM T59328 CV60ME 44321734 IC50 > 50000 nM T59328 C94MXP 44324651 IC50 = 170 nM T59328 CY48CU 44324654 IC50 = 430 nM T59328 C7T9RZ 44324666 IC50 = 730 nM T59328 CMP9D5 44324692 IC50 = 390 nM T59328 C9M3UO 44324693 IC50 = 11400 nM T59328 CB94OP 44324694 IC50 = 820 nM T59328 CI4P0C 44324869 IC50 = 300 nM T59328 CR5YP3 44324917 IC50 = 780 nM T59328 CSRW08 44324921 IC50 = 910 nM T59328 C7D6AQ 44324941 IC50 = 660 nM T59328 CL1QG5 44324942 IC50 = 10 nM T59328 CHKY38 44325074 IC50 = 27 nM T59328 CGHA16 44325116 IC50 = 65 nM T59328 CKC7R3 44330975 IC50 = 80500 nM T59328 CYT6F3 44330976 IC50 > 100000 nM T59328 CU58ZC 44331212 IC50 = 170 nM T59328 C2BSI9 44333736 IC50 = 3.3 nM T59328 C1KSW5 44335197 IC50 = 300 nM T59328 CB5J4A 44345182 IC50 = 4500 nM T59328 CW42OA 44345288 IC50 = 8709.64 nM T59328 C0A6IM 44345309 IC50 = 7943.28 nM T59328 CO9U4D 44345316 IC50 = 3400 nM T59328 C92MBY 44345327 IC50 = 3200 nM T59328 C5SMO1 44345334 IC50 = 48000 nM T59328 C57GUL 44345336 IC50 = 707.95 nM T59328 C09YJV 44345337 IC50 = 87000 nM T59328 CL73FP 44345342 IC50 = 15000 nM T59328 CCL45B 44345353 IC50 > 167000 nM T59328 CR5EL2 44345383 IC50 = 2000 nM T59328 CI02JL 44345396 IC50 = 4400 nM T59328 CHE2P1 44345431 IC50 = 900 nM T59328 CRQ76V 44345433 IC50 = 640 nM T59328 CJB1C4 44345439 IC50 = 5600 nM T59328 CVZ05R 44345469 IC50 = 6760.83 nM T59328 C0SH6O 44345633 IC50 = 14800 nM T59328 C06AQN 44345644 IC50 = 14454.4 nM T59328 CD62QG 44345647 IC50 = 5300 nM T59328 C2ESL8 44345648 IC50 = 12000 nM T59328 CW15XR 44345649 IC50 = 1700 nM T59328 CBC01N 44345675 IC50 > 50000 nM T59328 CPC35U 44345676 IC50 > 50000 nM T59328 C0KD4U 44346053 IC50 = 1100 nM T59328 CR1L3W 44346250 IC50 = 450000 nM T59328 C0D3UQ 44347328 IC50 = 9700 nM T59328 CJKU43 44347354 IC50 = 10300 nM T59328 C1QDI7 44347577 IC50 = 27200 nM T59328 C3WQ6J 44352770 IC50 = 910 nM T59328 C92FHZ 44352771 IC50 = 1300 nM T59328 CBX2L9 44352772 IC50 = 1100 nM T59328 CFJK28 44352785 IC50 = 7000 nM T59328 CF65DQ 44352791 IC50 > 100000 nM T59328 CL5QU9 44352816 IC50 = 3500 nM T59328 CKD32G 44352817 IC50 = 6400 nM T59328 CTZ3O4 44352818 IC50 = 1100 nM T59328 CRV1T2 44352826 IC50 = 160 nM T59328 CKGI05 44352842 IC50 = 110 nM T59328 C7YJ1S 44352843 IC50 = 7400 nM T59328 C8EVN3 44352844 IC50 = 3600 nM T59328 CI1R2S 44352845 IC50 > 70000 nM T59328 CQN85G 44352860 IC50 = 8180 nM T59328 CO43ND 44352873 IC50 = 13500 nM T59328 C2WRC4 44352890 IC50 = 4600 nM T59328 C1KO6C 44352905 IC50 = 12500 nM T59328 CK56AZ 44352914 IC50 = 4700 nM T59328 C2T4XV 44352915 IC50 = 8180 nM T59328 CX1SD9 44352928 IC50 = 2400 nM T59328 CIUR28 44352929 IC50 = 1300 nM T59328 CJE57B 44352930 IC50 = 4800 nM T59328 C84FIH 44352951 IC50 = 2600 nM T59328 CVHA74 44352970 IC50 = 260 nM T59328 CQ2F5D 44352972 IC50 = 17 nM T59328 CX82RD 44352973 IC50 = 220 nM T59328 COZ52V 44353100 IC50 = 31 nM T59328 CLX76Q 44353115 IC50 = 19 nM T59328 C9RUC6 44353122 IC50 = 330 nM T59328 CUG68J 44353130 IC50 = 43 nM T59328 C50EHA 44353341 IC50 > 100000 nM T59328 CP8B0J 44353452 IC50 > 100000 nM T59328 CQZM34 44355143 IC50 > 20000 nM T59328 CX1I0D 44355168 IC50 > 1000 nM T59328 C2F9DZ 44355323 IC50 > 20000 nM T59328 C4LKS3 44355443 IC50 = 100 nM T59328 CJWK61 44355456 IC50 > 50000 nM T59328 C9YI1R 44355486 IC50 = 10 nM T59328 CM0BW2 44355543 IC50 > 50000 nM T59328 C0VSJ3 44355545 IC50 > 20000 nM T59328 CIV6A3 44355618 IC50 = 12000 nM T59328 CYR4C8 44355673 IC50 > 50000 nM T59328 CM24OQ 44355891 IC50 > 20000 nM T59328 CHL4V6 44355892 IC50 > 20000 nM T59328 CM6X3O 44355907 IC50 = 1300 nM T59328 C30OUK 44355908 IC50 = 7000 nM T59328 CX0R3O 44355931 IC50 > 50000 nM T59328 CK4U5B 44361553 IC50 = 1698.24 nM T59328 CM56JY 44361640 IC50 = 3019.95 nM T59328 CT2R7Z 44361668 IC50 = 15848.93 nM T59328 C5RZI9 44361703 IC50 = 19054.61 nM T59328 C04PXM 44361706 IC50 = 47863.01 nM T59328 C1NRF6 44361710 IC50 = 53703.18 nM T59328 CAZD14 44361915 IC50 = 165958.69 nM T59328 CFY75E 44363476 IC50 = 2100 nM T59328 C1FM7A 44367247 IC50 = 2.7 nM T59328 CSW63A 44367400 IC50 > 10000 nM T59328 CWJ61S 44367436 IC50 = 33 nM T59328 C0RBE5 44367446 IC50 = 85 nM T59328 CQL29S 44367457 IC50 = 9.4 nM T59328 C9GX4S 44367566 IC50 = 40 nM T59328 CYV2D7 44368815 IC50 > 10000 nM T59328 C10VDK 44371971 IC50 = 330 nM T59328 C2GRI5 44372004 IC50 = 10 nM T59328 C9NYG0 44372005 IC50 = 110 nM T59328 CFM6C8 44372022 IC50 = 8 nM T59328 CCGX21 44372180 IC50 = 35 nM T59328 C6L4CX 44372197 IC50 = 82 nM T59328 CSA68M 44372283 IC50 = 540 nM T59328 C8RL0S 44377259 IC50 = 3.9 nM T59328 CC3T6E 44381073 IC50 = 13200 nM T59328 CQT59Y 44381095 IC50 = 9700 nM T59328 C8LZ0Q 44381185 IC50 = 600 nM T59328 C6FCU8 44381190 IC50 = 440 nM T59328 C1D2LU 44381191 IC50 = 830 nM T59328 CJZD30 44381192 IC50 = 740 nM T59328 CFQ57C 44381224 IC50 = 570 nM T59328 CZ64TC 44381237 IC50 = 80 nM T59328 C5WQY2 44381238 IC50 = 250 nM T59328 CD0WU4 44381266 IC50 = 420 nM T59328 C7VJ9M 44381267 IC50 = 2820 nM T59328 C9S1EJ 44381268 IC50 = 790 nM T59328 CM64RL 44381269 IC50 = 300 nM T59328 CBKP57 44381381 IC50 = 450 nM T59328 C2DCJ0 44381398 IC50 = 8300 nM T59328 C6LSB4 44381409 IC50 = 295 nM T59328 CE7H4L 44381435 IC50 = 500 nM T59328 C98OGL 44381436 IC50 = 330 nM T59328 CEQ7M0 44381445 IC50 = 930 nM T59328 CWKB67 44381507 IC50 = 14400 nM T59328 CX98KS 44381508 IC50 = 440 nM T59328 C6LC8M 44381556 IC50 = 310 nM T59328 CCA56B 44381571 IC50 = 1470 nM T59328 C5Z9MJ 44381580 IC50 = 750 nM T59328 CY58LS 44381608 IC50 = 2100 nM T59328 C6DQX7 44381674 IC50 = 2200 nM T59328 C75NGL 44384514 IC50 = 1300 nM T59328 CV0F4D 44384547 IC50 = 12000 nM T59328 CQF8Y7 44384548 IC50 = 1100 nM T59328 CF01AV 44384717 IC50 = 5300 nM T59328 CI2L9R 44384964 IC50 = 6400 nM T59328 CC09FT 44384965 IC50 = 1400 nM T59328 CE9PU7 44385035 IC50 = 6400 nM T59328 CQGW07 44385080 IC50 = 700 nM T59328 CL4Y9M 44385116 IC50 = 800 nM T59328 CUI34C 44385739 IC50 = 2650 nM T59328 C87MAJ 44388483 IC50 = 72 nM T59328 CB7QM3 44388486 IC50 = 151 nM T59328 C6WDG3 44388487 IC50 = 210 nM T59328 C3YM9F 44388494 IC50 = 255 nM T59328 CN4L2V 44388499 IC50 = 247 nM T59328 CUA90G 44388501 IC50 = 400 nM T59328 CBU34A 44389468 IC50 = 26 nM T59328 CU9Z5Y 44395043 IC50 = 490 nM T59328 CF31XZ 44395044 IC50 > 33000 nM T59328 CCLX29 44395123 IC50 = 2800 nM T59328 CCAI71 44395145 IC50 > 33000 nM T59328 CZ97PV 44395162 IC50 = 2200 nM T59328 CZ6HP1 44395171 IC50 = 11000 nM T59328 C2T6DH 44395178 IC50 = 29000 nM T59328 C0XQ2Z 44395209 IC50 > 33000 nM T59328 CTDI68 44395241 IC50 > 33000 nM T59328 CW3BP8 44398371 IC50 = 45800 nM T59328 CH9NR8 44403081 IC50 = 200 nM T59328 C0AR9C 44403420 IC50 = 5 nM T59328 CGQ26K 44403425 IC50 = 1800 nM T59328 CRV6B4 44403429 IC50 = 2400 nM T59328 CTY5K7 44403435 IC50 = 2100 nM T59328 C47XFZ 44403436 IC50 = 440 nM T59328 C8K4AL 44407237 IC50 = 12600 nM T59328 CUA18B 44407238 IC50 = 31000 nM T59328 C04HFE 44407248 IC50 > 50000 nM T59328 CR3O1C 44407275 IC50 = 5100 nM T59328 C70BFV 44407276 IC50 = 13600 nM T59328 CMH7W6 44407277 IC50 = 9000 nM T59328 CIQR47 44409038 IC50 = 1700 nM T59328 C6UE2S 44409043 IC50 = 3700 nM T59328 C64ZYA 44409055 IC50 = 3400 nM T59328 CY1AQ7 44409056 IC50 = 7000 nM T59328 CT9M4U 44409118 IC50 = 873 nM T59328 C46NPW 44409144 IC50 = 225 nM T59328 C6E4QU 44409147 IC50 = 1000 nM T59328 C29RFN 44409148 IC50 = 9601 nM T59328 C9H3VZ 44409149 IC50 = 671 nM T59328 C4V6FS 44409152 IC50 > 10000 nM T59328 CW24DU 44409153 IC50 = 5400 nM T59328 C4S6ZN 44409156 IC50 = 4900 nM T59328 C3HFY0 44409208 IC50 = 3 nM T59328 CW87XM 44409211 IC50 = 66 nM T59328 CHD92U 44409225 IC50 = 2000 nM T59328 CNS1X6 44409226 IC50 = 9800 nM T59328 CIX8D6 44409229 IC50 > 10000 nM T59328 C2MN0X 44409230 IC50 > 10000 nM T59328 CNQL75 44409263 IC50 = 1000 nM T59328 C7G6OS 44409281 IC50 > 10000 nM T59328 C0TNV5 44409288 IC50 < 2 nM T59328 C8UN1W 44409346 IC50 = 1000 nM T59328 CQW9E1 44409347 IC50 = 10 nM T59328 C03UCB 44409353 IC50 = 4400 nM T59328 C7W8VG 44409387 IC50 = 1384 nM T59328 C9SP0E 44409388 IC50 < 2 nM T59328 CM1D9O 44409422 IC50 = 187 nM T59328 CZQ03C 44409423 IC50 = 8068 nM T59328 C7HD4Q 44410411 IC50 = 320 nM T59328 CED5S6 44410414 IC50 = 85 nM T59328 C0A7XB 44410560 IC50 = 63 nM T59328 C5WKG0 44410574 IC50 = 25100 nM T59328 CDQ4S6 44410648 IC50 = 42 nM T59328 C4OJ1S 44410700 IC50 = 110 nM T59328 CIY53K 44410704 IC50 = 79 nM T59328 CPH17L 44410710 IC50 = 50 nM T59328 C2J1KU 44410716 IC50 = 31 nM T59328 CV09DY 44410717 IC50 = 8 nM T59328 CP3CI1 44410720 IC50 = 50 nM T59328 C8W7AD 44410723 IC50 = 40 nM T59328 CAT5X4 44410829 IC50 = 300 nM T59328 CC6Y5P 44410844 IC50 = 300 nM T59328 CG34TY 44410851 IC50 = 70 nM T59328 C41EIA 44410869 IC50 = 10 nM T59328 CB6AE8 44410948 IC50 = 70 nM T59328 CXZG12 44410949 IC50 < 1 nM T59328 CS7IE9 44410953 IC50 = 100 nM T59328 CA9M4X 44410954 IC50 = 90 nM T59328 C3SP5H 44410955 IC50 = 450 nM T59328 C5D6YP 44410956 IC50 = 10 nM T59328 C5W1VC 44410959 IC50 = 130 nM T59328 CM1C2G 44410960 IC50 = 30 nM T59328 CVSI80 44411048 IC50 = 80 nM T59328 CN72BR 44411161 IC50 = 50 nM T59328 C4AW0O 44411183 IC50 = 25 nM T59328 C0XJC3 44412177 IC50 = 1693 nM T59328 C5QD2S 44412181 IC50 = 81 nM T59328 CRH3Y6 44412244 IC50 = 156 nM T59328 C7KZV2 44414322 IC50 > 50000 nM T59328 CJM06T 44414347 IC50 > 50000 nM T59328 C16IVC 44416188 IC50 = 50 nM T59328 COFI73 44416243 IC50 = 16 nM T59328 CS8U4Y 44416288 IC50 = 19 nM T59328 CVA3S4 44416289 IC50 = 17 nM T59328 CD4H3O 44416334 IC50 = 62900 nM T59328 CO25JT 44416335 IC50 = 14100 nM T59328 C1KW2L 44416347 IC50 > 100000 nM T59328 CMG28W 44416407 IC50 = 51 nM T59328 C5R7IW 44416429 IC50 = 7400 nM T59328 C7C4TK 44416433 IC50 = 6100 nM T59328 C0IUL9 44416434 IC50 = 4600 nM T59328 CUBA46 44416461 IC50 = 18 nM T59328 CR42NY 44416467 IC50 = 10800 nM T59328 C5XE7I 44416473 IC50 = 15200 nM T59328 CAP9S0 44416499 IC50 = 24600 nM T59328 C41SAP 44416508 IC50 = 3400 nM T59328 CA83EK 44416509 IC50 = 8200 nM T59328 CK8R2O 44416545 IC50 = 1200 nM T59328 CX17JM 44416560 IC50 = 150 nM T59328 CD2FC0 44416568 IC50 = 5600 nM T59328 CPIA51 44416569 IC50 > 100000 nM T59328 C7QH2K 44416595 IC50 = 114 nM T59328 CX3DU9 44416596 IC50 > 100000 nM T59328 CYU1W9 44416603 IC50 = 17000 nM T59328 C7DTI2 44416610 IC50 < 0.5 nM T59328 CJS8C5 44416611 IC50 = 9 nM T59328 C0CQ4S 44416612 IC50 = 1 nM T59328 C35BCH 44416635 IC50 = 300 nM T59328 CO9MX1 44416647 IC50 = 14500 nM T59328 C6HQ5D 44416655 IC50 = 1100 nM T59328 CIY3J4 44416673 IC50 = 9 nM T59328 CIV18H 44416687 IC50 = 300 nM T59328 C43VZI 44416688 IC50 = 800 nM T59328 CF5UH3 44416692 IC50 = 900 nM T59328 C43NYR 44416693 IC50 = 8700 nM T59328 C8RHO3 44416712 IC50 = 200 nM T59328 C2L0ZB 44416719 IC50 = 106 nM T59328 CZ3WQ2 44416741 IC50 = 7100 nM T59328 CAV3B1 44417449 IC50 > 3000 nM T59328 CKD97C 44417487 IC50 > 3000 nM T59328 COPG94 44427519 IC50 > 10000 nM T59328 C0PLD7 44428887 IC50 = 283.3 nM T59328 C2V1FP 44428888 IC50 = 43.1 nM T59328 C2UT9G 44428889 IC50 = 166.7 nM T59328 C8XRO1 44428890 IC50 = 18.7 nM T59328 C3A2HC 44428891 IC50 = 791.9 nM T59328 C42KHG 44428893 IC50 = 35.6 nM T59328 CDE73U 44428895 IC50 = 295.2 nM T59328 C5H3DV 44428898 IC50 = 107.3 nM T59328 C2V1ER 44428899 IC50 = 173.1 nM T59328 CLGZ52 44428901 IC50 < 10 nM T59328 C8LI7S 44428906 IC50 = 7710 nM T59328 C7BZ0K 44430019 IC50 = 81 nM T59328 CJ1U9R 44430027 IC50 = 1000 nM T59328 COBA27 44430030 IC50 = 140 nM T59328 C8WJV9 44430032 IC50 = 130 nM T59328 C9UYP5 44430034 IC50 = 26 nM T59328 CQ67VA 44430037 IC50 = 190 nM T59328 CW58IO 44430039 IC50 = 130 nM T59328 CA98KR 44432441 IC50 > 6000 nM T59328 C5QJ0K 44435405 IC50 < 5000 nM T59328 CNSW23 44435406 IC50 > 40000 nM T59328 CIOY17 44435407 IC50 > 40000 nM T59328 CCV5A0 44435408 IC50 > 40000 nM T59328 C73EMA 44435409 IC50 > 40000 nM T59328 CAJ5W6 44435435 IC50 > 40000 nM T59328 CX09ZA 44440812 IC50 = 210 nM T59328 C36FXV 44440815 IC50 = 86 nM T59328 CF5UR8 44440816 IC50 = 200 nM T59328 C87FRB 44440817 IC50 = 1800 nM T59328 CNCU91 44440820 IC50 = 340 nM T59328 CL1N3P 44440821 IC50 = 490 nM T59328 C85SOF 44440823 IC50 = 30 nM T59328 C8GHB0 44440824 IC50 = 460 nM T59328 C74ONA 44440826 IC50 = 140 nM T59328 CNU0P1 44440830 IC50 = 130 nM T59328 CU72VL 44440831 IC50 = 190 nM T59328 CNY07A 44440833 IC50 = 83 nM T59328 CZ4G2C 44440835 IC50 = 640 nM T59328 C85HCV 44440836 IC50 = 210 nM T59328 CO6DP3 44440837 IC50 = 560 nM T59328 C4Y1TD 44440839 IC50 = 500 nM T59328 CWC9V6 44440840 IC50 = 810 nM T59328 CIF14K 44440841 IC50 = 120 nM T59328 CJ23DP 44440842 IC50 = 690 nM T59328 CO8WZ7 44440843 IC50 = 68 nM T59328 CJL0G8 44440844 IC50 = 400 nM T59328 CA75PM 44440874 IC50 = 430 nM T59328 CAM78I 44441000 IC50 = 50 nM T59328 C6ZEJ5 44441012 IC50 = 190 nM T59328 C3MW6G 44441013 IC50 = 40 nM T59328 C3AZF8 44441014 IC50 = 47 nM T59328 CJC06N 44441015 IC50 = 190 nM T59328 CWJ1U3 44441016 IC50 = 530 nM T59328 C2IL0Y 44441017 IC50 = 19 nM T59328 CMW7T5 44442025 IC50 = 3 nM T59328 C3U1GC 44442026 IC50 = 2580 nM T59328 C9J2FM 44442027 IC50 = 2 nM T59328 CU7N0D 44442028 IC50 = 191 nM T59328 C8OSC2 44442129 IC50 = 331 nM T59328 CN0PD8 44442133 IC50 = 1640.6 nM T59328 CH4T0Y 44442137 IC50 = 185.8 nM T59328 CX2F5J 44442142 IC50 = 114.2 nM T59328 C4LNA9 44442145 IC50 = 94.5 nM T59328 CLD6A1 44442146 IC50 = 151.5 nM T59328 CKBP38 44442147 IC50 = 50.3 nM T59328 CDT1F0 44442149 IC50 = 88.7 nM T59328 C5ETZ9 44442150 IC50 = 921 nM T59328 CZKI61 44442152 IC50 = 402.1 nM T59328 CC06RB 44442154 IC50 = 1362.6 nM T59328 CGY4Q2 44442155 IC50 = 205.8 nM T59328 C8CIJ2 44442169 IC50 = 13 nM T59328 C36JSL 44442170 IC50 = 80 nM T59328 CD3LW7 44442179 IC50 = 4 nM T59328 C8LY2G 44442184 IC50 = 10 nM T59328 CPQ02C 44442185 IC50 = 12 nM T59328 CGFL71 44442186 IC50 = 1.8 nM T59328 CEX85R 44442187 IC50 = 11.7 nM T59328 CY61BH 44442188 IC50 = 4.2 nM T59328 C5JRD8 44442189 IC50 = 662 nM T59328 C5R4QE 44442729 Ki = 24 nM T59328 CGC76I 44442730 Ki = 180 nM T59328 CJM6N5 44442731 Ki = 360 nM T59328 CH2FS6 44442732 Ki = 120 nM T59328 CZ7FC6 44442733 Ki = 64 nM T59328 C6PNZ4 44442734 Ki = 52 nM T59328 C8N1EQ 44442735 Ki = 68 nM T59328 C26EVP 44442736 IC50 = 173 nM T59328 C0S6PN 44442737 IC50 = 52.8 nM T59328 CAZ5O7 44442738 IC50 = 5 nM T59328 CM9XW1 44442739 Ki = 360 nM T59328 CFOH51 44442740 Ki = 340 nM T59328 CX10DZ 44442742 Ki = 40 nM T59328 CN12IA 44442744 Ki = 400 nM T59328 C0DOP6 44442745 Ki = 80 nM T59328 CJ4BV0 44442747 Ki = 44 nM T59328 CJHV89 44442752 Ki = 80 nM T59328 CYS18W 44442753 Ki = 220 nM T59328 C26GVA 44442758 Ki = 52 nM T59328 CZG61W 44442759 Ki = 36 nM T59328 C4YMI9 44447890 IC50 > 1000 nM T59328 CR65PM 44447895 IC50 > 1000 nM T59328 CR62KV 44448938 IC50 = 267 nM T59328 CT9R7H 44448969 IC50 = 306 nM T59328 C9RV4Q 44448995 IC50 = 1123 nM T59328 CUB12D 44449577 IC50 = 150 nM T59328 CSA12W 44450544 IC50 = 5000000 nM T59328 C3ZBV8 44450546 IC50 = 13300 nM T59328 C0C2RS 44450792 IC50 = 780 nM T59328 C0MXV2 44450803 IC50 > 10000 nM T59328 C7HIM2 44452543 IC50 > 500 nM T59328 CZ9H4D 44452544 IC50 > 500 nM T59328 CQ1M7K 44455194 IC50 < 1 nM T59328 C86DQE 44455195 IC50 = 28 nM T59328 C20ISD 44455293 IC50 = 13 nM T59328 CUN90T 44455330 IC50 = 18 nM T59328 CNR2V1 44456900 IC50 = 3.236 nM T59328 C3AWN6 44456909 IC50 = 1.514 nM T59328 CBD75X 44456910 IC50 = 40.74 nM T59328 CAM6P8 44456911 IC50 = 4786.3 nM T59328 CVYZ16 44456912 IC50 = 3715.35 nM T59328 C7GQR6 44456927 IC50 = 0.912 nM T59328 C6S5YU 44456928 IC50 = 8.511 nM T59328 CHE0Q7 44456929 IC50 = 25.7 nM T59328 C7J4MG 44456940 IC50 = 0.5129 nM T59328 CD18RN 44456941 IC50 = 245.47 nM T59328 CIWS70 44456942 IC50 = 10 nM T59328 C1MI8R 44456962 IC50 = 7.413 nM T59328 C3P2SB 44456963 IC50 = 40.74 nM T59328 CAF3L1 44456987 IC50 = 7.244 nM T59328 CLW80I 44456989 IC50 = 251.19 nM T59328 CF1UQ0 44457004 IC50 = 45.71 nM T59328 C93BJI 44457005 IC50 = 8.913 nM T59328 CJB04A 44457006 IC50 = 39.81 nM T59328 C7B2RU 44457007 IC50 = 13.18 nM T59328 CAF6E5 44457023 IC50 = 12.02 nM T59328 C7FE2H 44457024 IC50 = 1.202 nM T59328 CVB57O 44457026 IC50 = 3.236 nM T59328 C8K3BG 44457027 IC50 = 14.13 nM T59328 C5MFW9 44457038 IC50 = 0.9333 nM T59328 C0R5SP 44457039 IC50 = 0.2455 nM T59328 C9XD8N 44457040 IC50 = 2.63 nM T59328 C8I0UN 44457041 IC50 = 29.51 nM T59328 CDK0Q7 44457055 IC50 = 9.333 nM T59328 C0P7JH 44457062 IC50 = 3.548 nM T59328 CQF2J4 44457064 IC50 = 9.333 nM T59328 C3JX0B 44457065 IC50 = 5.623 nM T59328 C8ZG4J 44457066 IC50 = 5.495 nM T59328 CB7Z4F 44457080 IC50 = 1.413 nM T59328 C2R4QL 44457083 IC50 = 16.22 nM T59328 C5G2UO 44457084 IC50 = 0.2818 nM T59328 C24HUL 44457085 IC50 = 2.344 nM T59328 C63CIA 44457086 IC50 = 5.012 nM T59328 CI39XF 44457115 IC50 = 5.495 nM T59328 CR06HM 44457116 IC50 = 40.74 nM T59328 CDV1E5 44457117 IC50 = 120.23 nM T59328 C5Y7HJ 44457118 IC50 = 70.79 nM T59328 C1PWV8 44457132 IC50 = 0.6166 nM T59328 C62QBG 44457133 IC50 = 1.905 nM T59328 C49BNA 44457135 IC50 = 4897.79 nM T59328 C35NVA 44457136 IC50 = 851.14 nM T59328 C9FMH7 44457137 IC50 = 1819.7 nM T59328 CU1I4O 44457148 IC50 = 676.08 nM T59328 CZ1R3H 44457149 IC50 = 131.83 nM T59328 CL0P5W 44471009 IC50 = 0.22 nM T59328 CAS03E 44481081 IC50 = 1340 nM T59328 C4TF5E 44481332 IC50 = 1760 nM T59328 C9D2SF 44515230 IC50 = 270 nM T59328 C5RA7I 44515232 IC50 = 850 nM T59328 CYH6P3 44520205 IC50 = 2090 nM T59328 CDFI53 44528870 IC50 = 68 nM T59328 CI8X2C 44528924 IC50 = 4 nM T59328 C9ZU2D 44528930 IC50 = 138 nM T59328 CXR98Y 44528960 IC50 = 6 nM T59328 CI3JR0 44532526 IC50 > 50000 nM T59328 CFP97X 44532811 IC50 = 3 nM T59328 C0LY6E 44552561 EC50 > 10000 nM T59328 C7KRU3 44552562 IC50 > 10000 nM T59328 CRPM76 44555376 IC50 = 200 nM T59328 C3JUM4 44555383 IC50 = 630 nM T59328 CYV71I 44555430 IC50 = 15.5 nM T59328 C3VRO9 44557921 IC50 > 10000 nM T59328 C1A4XG 44562420 IC50 = 458 nM T59328 C3UV2W 44562431 IC50 = 620 nM T59328 C5AS8P 44564023 IC50 = 1.514 nM T59328 CA8E5X 44564024 IC50 = 19.95 nM T59328 C68VDI 44564025 IC50 = 6.607 nM T59328 CPO8W9 44564026 IC50 = 0.912 nM T59328 C1K6BV 44564031 IC50 = 0.1698 nM T59328 CYE06Q 44564061 IC50 = 1.585 nM T59328 C93BFU 44564062 IC50 = 1.202 nM T59328 CLAF15 44564063 IC50 = 0.5012 nM T59328 C2T8PE 44564064 IC50 = 0.5495 nM T59328 CX2Q1J 44564065 IC50 = 0.6918 nM T59328 CX4M3C 44564100 IC50 = 1.738 nM T59328 COSJ65 44564101 IC50 = 1.096 nM T59328 CLYD65 44564102 IC50 = 1.585 nM T59328 C9BA2G 44564103 IC50 = 9.12 nM T59328 CD5QH9 44564104 IC50 = 1.202 nM T59328 C8G6MO 44564165 IC50 = 0.7079 nM T59328 CIW9B5 44564166 IC50 = 44.67 nM T59328 CN4WY6 44564167 IC50 = 26.92 nM T59328 CN0AS3 44564168 IC50 = 0.3715 nM T59328 C59GKR 44564169 IC50 = 2.692 nM T59328 CW13TY 44564170 IC50 = 1.514 nM T59328 CC17KX 44564171 IC50 = 4.169 nM T59328 CX0US9 44564172 IC50 = 2.692 nM T59328 C0TUR8 44564191 IC50 = 3.311 nM T59328 CD45HS 44564192 IC50 = 2.399 nM T59328 C4VQP9 44564193 IC50 = 0.4365 nM T59328 C81WPX 44564194 IC50 = 1.096 nM T59328 COQ61X 44564233 IC50 = 0.7244 nM T59328 C0Y2WH 44564234 IC50 = 0.8128 nM T59328 CPLB92 44564235 IC50 = 0.5623 nM T59328 C1KWB4 44564236 IC50 = 1.445 nM T59328 C04JAC 44564270 IC50 = 93.33 nM T59328 C9VAI7 44564303 IC50 = 0.4467 nM T59328 CXI08J 44564304 IC50 = 0.537 nM T59328 C2DS5N 44564306 IC50 = 8.6 nM T59328 CM3J7B 44564307 IC50 = 6 nM T59328 CP9RO4 44564308 IC50 = 8 nM T59328 CF41OU 44564309 IC50 = 8 nM T59328 CQ0ID4 44564335 IC50 < 1 nM T59328 CAE13O 44564361 IC50 = 1.096 nM T59328 C59TUM 44564362 IC50 = 1.202 nM T59328 C4ZTX0 44564365 IC50 = 10320 nM T59328 C1QFI4 44564394 IC50 = 1.698 nM T59328 CZCF57 44564395 IC50 = 3.631 nM T59328 CXFP58 44564396 IC50 = 3.89 nM T59328 C5VO9D 44564397 IC50 = 3.02 nM T59328 C29OUL 44564398 IC50 = 3.715 nM T59328 CFU1Q8 44564399 IC50 = 0.4365 nM T59328 CD10EC 44564400 IC50 = 5390 nM T59328 CF1T5K 44564401 IC50 = 13570 nM T59328 CD6XJ4 44564402 IC50 = 5220 nM T59328 C7OU0D 44564403 IC50 = 10590 nM T59328 CYD0K8 44564435 IC50 = 0.7762 nM T59328 CS92EV 44564436 IC50 = 0.4169 nM T59328 C41PEW 44564437 IC50 = 1.995 nM T59328 C4CH2U 44564438 IC50 = 1.514 nM T59328 C58LAW 44564439 IC50 = 0.6918 nM T59328 C27UGT 44564440 IC50 = 0.7943 nM T59328 CNQE26 44564441 IC50 = 1.585 nM T59328 C8UR0S 44564442 IC50 = 40.74 nM T59328 CZ1LX2 44564443 IC50 = 20.89 nM T59328 C2PTY9 44564444 IC50 = 3.715 nM T59328 C6NB0I 44564445 IC50 = 7500 nM T59328 CLR6X7 44564476 IC50 = 1.82 nM T59328 CEUJ39 44564477 IC50 = 0.7586 nM T59328 COR0K6 44564478 IC50 = 1.514 nM T59328 C5P0CL 44564479 IC50 = 1.698 nM T59328 CV67XP 44564480 IC50 = 8.71 nM T59328 CO6C8D 44564481 IC50 = 5.129 nM T59328 C91WOF 44564482 IC50 = 4.786 nM T59328 CB1O0P 44564526 IC50 = 0.7586 nM T59328 C4T3PW 44564527 IC50 = 0.1585 nM T59328 CR2J8L 44564528 IC50 = 2.692 nM T59328 C3NMY1 44564529 IC50 = 0.955 nM T59328 CXD0W8 44564530 IC50 = 0.9772 nM T59328 CC62JT 44564704 IC50 = 150 nM T59328 CC7E4K 44564705 IC50 > 10000 nM T59328 C42ZEW 44564706 IC50 = 2000 nM T59328 C53MCK 44564747 IC50 > 10000 nM T59328 CDI31F 44564748 IC50 > 10000 nM T59328 CA17NT 44564749 IC50 > 10000 nM T59328 CMIZ20 44564750 IC50 > 10000 nM T59328 CSO9F8 44564751 IC50 > 10000 nM T59328 C8ATG9 44564787 IC50 > 10000 nM T59328 CM50GS 44564788 IC50 > 10000 nM T59328 C3Q0DX 44564789 IC50 = 1300 nM T59328 CP40XB 44564790 IC50 = 720 nM T59328 C35NTB 44564791 IC50 = 7700 nM T59328 CJY83G 44564817 IC50 = 5100 nM T59328 CLK98G 44564818 IC50 = 7800 nM T59328 CF2D1K 44564819 IC50 = 2600 nM T59328 C3CQ9K 44564820 IC50 > 10000 nM T59328 CI8V2L 44564821 IC50 > 10000 nM T59328 C9PO7J 44564860 IC50 > 10000 nM T59328 C16FJW 44564861 IC50 > 10000 nM T59328 C8AMX5 44564862 IC50 = 5300 nM T59328 CTR59U 44564863 IC50 > 10000 nM T59328 C9EY4C 44564864 IC50 = 800 nM T59328 CG5Z7T 44564910 IC50 > 10000 nM T59328 CU9O4C 44564911 IC50 > 10000 nM T59328 CXZ15S 44564954 IC50 > 10000 nM T59328 CZ78WJ 44564955 IC50 > 10000 nM T59328 CJ1X9V 44565013 IC50 = 1900 nM T59328 CN2Q3D 44565014 IC50 = 3300 nM T59328 CM2GN3 44565015 IC50 > 10000 nM T59328 C6RV9I 44565016 IC50 = 1700 nM T59328 CJC85A 44565069 IC50 = 1600 nM T59328 CSOH56 44565943 IC50 > 200000 nM T59328 CTUD59 44565958 IC50 > 200000 nM T59328 C6IFZ9 44565965 IC50 > 200000 nM T59328 CRX0M5 44571414 IC50 = 304 nM T59328 C9KY2N 44571415 IC50 = 115 nM T59328 CT92ZI 44571431 IC50 = 10 nM T59328 C0W9NE 44571432 IC50 = 4 nM T59328 CKY57M 44571433 IC50 = 8 nM T59328 C2RQ3H 44571434 IC50 = 7 nM T59328 CUCI91 44571435 IC50 = 15 nM T59328 C7LVG6 44571436 IC50 = 54 nM T59328 CIU14N 44571437 IC50 = 121 nM T59328 CLP71D 44571448 IC50 = 2 nM T59328 CEIK76 44571449 IC50 = 5 nM T59328 CFNT92 44571450 IC50 = 3 nM T59328 CIB7R5 44571451 IC50 = 3 nM T59328 CK6L2W 44571452 IC50 = 68 nM T59328 CI1PL5 44571453 IC50 = 9 nM T59328 CZ0ID1 44571454 IC50 = 96 nM T59328 CWFB42 44571820 IC50 = 22 nM T59328 CU9Y0V 44576127 IC50 = 0.9 ug.mL-1 T59328 CPKL09 44576144 IC50 = 800 nM T59328 CG4E2Z 44576145 IC50 = 600 nM T59328 CI87PR 44576146 IC50 = 3000 nM T59328 C2U7IW 44576150 IC50 = 6000 nM T59328 C8ST7I 44576151 IC50 = 900000 nM T59328 C3K5AT 44576152 IC50 = 10000 nM T59328 CI8J1E 44576153 IC50 = 10000 nM T59328 CD0AC6 44576154 IC50 = 400000 nM T59328 C35DJE 44576155 IC50 = 600000 nM T59328 C9YXF6 44576156 IC50 = 600000 nM T59328 C4KBE3 44576157 IC50 = 1000 nM T59328 CQL4X2 44576163 IC50 = 10000 nM T59328 C7Q1VU 44580077 IC50 > 25000 nM T59328 CL90SE 44580358 IC50 > 25000 nM T59328 CK1VE7 44580420 IC50 > 25000 nM T59328 CH2R7X 44580449 IC50 > 25000 nM T59328 C1VH0C 44580532 IC50 > 25000 nM T59328 CXC52J 44580649 IC50 > 25000 nM T59328 CE32BQ 44580689 IC50 = 700 nM T59328 C8Z5AX 44580778 IC50 > 25000 nM T59328 C9XIA1 44580891 IC50 = 109 nM T59328 CZC2R9 44580892 IC50 = 130 nM T59328 CYSF35 44580915 IC50 = 120 nM T59328 CP81ZN 44580916 IC50 = 58 nM T59328 CQL7G0 44580917 IC50 = 140 nM T59328 C8LK3H 44580918 IC50 = 14 nM T59328 C5H1XE 44580949 IC50 = 115 nM T59328 C2I8SC 44580950 IC50 = 81 nM T59328 CK9NC7 44580951 IC50 = 63 nM T59328 CO6A7L 44580971 IC50 = 141 nM T59328 CHSR02 44581016 IC50 = 60 nM T59328 C06LHO 44581017 IC50 = 50 nM T59328 CQV6W9 44586019 IC50 = 670 nM T59328 C5WOE2 44586449 IC50 = 300 nM T59328 C0VF8M 44586450 IC50 = 2200 nM T59328 C4K7NP 44586451 IC50 = 3400 nM T59328 C1JNR5 44586452 IC50 = 4700 nM T59328 C6T8UP 44586490 IC50 = 22800 nM T59328 CU95NI 44586526 IC50 > 200000 nM T59328 CBK9R3 44586527 IC50 = 1320 nM T59328 CA18IW 44586528 IC50 = 3180 nM T59328 C0YSZ2 44586577 IC50 > 200000 nM T59328 CTHK89 44587526 IC50 = 49 nM T59328 C7BP3R 44587569 IC50 = 9 nM T59328 CXN7Z2 44592167 IC50 = 82 nM T59328 CM16KD 44592210 IC50 = 7 nM T59328 C6OZB8 44592211 IC50 = 10 nM T59328 C9NXT5 44592212 IC50 = 9 nM T59328 C70GPR 44592213 IC50 = 14 nM T59328 CKC47E 44592253 IC50 = 59 nM T59328 CZW9G8 44592254 IC50 = 17900 nM T59328 CQKV92 44592255 IC50 = 27 nM T59328 C3XAR9 44592374 IC50 = 11 nM T59328 CL2Z5Q 44592375 IC50 = 6 nM T59328 COY57J 44592504 IC50 = 10000 nM T59328 C3M0SR 44593598 IC50 = 0.01 ug.mL-1 T59328 C70VZY 44593599 IC50 = 0.2 ug.mL-1 T59328 C6OC4Z 44607530 IC50 < 0.5 nM T59328 C8M5KI 44611919 IC50 = 68.2 nM T59328 C1EM3P 44629538 IC50 < 1 nM T59328 C2SHM5 44723861 IC50 = 3740 nM T59328 CJ2L1M 44820629 IC50 = 2200 nM T59328 CP2YM3 45103907 IC50 = 2400 nM T59328 C13CJG 45139788 IC50 = 1400 nM T59328 CD78OC 45139973 IC50 = 600 nM T59328 CU3RF1 45139989 IC50 > 10000 nM T59328 CQGZ06 45139991 IC50 > 10000 nM T59328 CXR3J0 45140149 IC50 = 28.8 nM T59328 C42EAO 45140150 IC50 = 1.99 nM T59328 CQ0WZ2 45140151 IC50 = 15.4 nM T59328 CCLE50 45140153 IC50 = 99.4 nM T59328 C4QVP3 45140347 IC50 = 268 nM T59328 CR8GN7 45140348 IC50 = 5077 nM T59328 C6K1JW 45140349 IC50 = 12.8 nM T59328 C82WLQ 45140350 IC50 = 125.6 nM T59328 CR4C9A 45140351 IC50 = 614 nM T59328 CB43GO 45141138 IC50 = 1.24 nM T59328 C61XCE 45141139 IC50 = 9.25 nM T59328 C4TEA9 45141140 IC50 = 291 nM T59328 C7YI9T 45141141 IC50 = 23.6 nM T59328 C47QIR 45141349 IC50 = 0.17 nM T59328 CTDP02 45141350 IC50 = 0.36 nM T59328 CU4RX5 45141351 IC50 = 0.85 nM T59328 C94WSQ 45141352 IC50 = 129 nM T59328 C8I4EW 45141586 IC50 = 0.37 nM T59328 CR4P3U 45151149 IC50 = 7480 nM T59328 C7W3UH 45151160 IC50 = 4680 nM T59328 C8C3JW 45151163 IC50 = 5710 nM T59328 CRM6V8 45151173 IC50 = 5070 nM T59328 CU29PK 45151176 IC50 = 4940 nM T59328 C0O6UA 45151186 IC50 = 7780 nM T59328 C8UGV5 45151203 IC50 = 6920 nM T59328 C6F8UE 45261965 IC50 = 350 nM T59328 C0T2MQ 45262036 IC50 = 4 nM T59328 CO28YF 45262447 IC50 = 20 nM T59328 CC31AL 45262457 IC50 > 100000 nM T59328 C5G9AS 45262479 IC50 = 444 nM T59328 C4DT3N 45262482 IC50 = 11 nM T59328 CC6RQ4 45262483 IC50 = 58 nM T59328 C87GSB 45262544 IC50 = 12.3 nM T59328 CX90FV 45265311 IC50 = 0.47 nM T59328 C2E3BZ 45265326 IC50 = 48 nM T59328 CO76KT 45265373 IC50 = 12.6 nM T59328 C56FXL 45265376 IC50 = 158 nM T59328 C5R3XP 45265596 IC50 = 460 nM T59328 C4DK0O 45265630 IC50 > 10000 nM T59328 CIX15N 45266023 IC50 = 120.23 nM T59328 CI82UE 45270897 IC50 > 10000 nM T59328 CKNP14 45276457 IC50 > 100000 nM T59328 CA4T0D 45276458 IC50 > 100000 nM T59328 C9BQM3 45370166 IC50 = 24 nM T59328 C6E2SC 45482700 IC50 > 10000 nM T59328 CZXH74 45482750 IC50 > 10000 nM T59328 CB6X7D 45483674 IC50 = 23 nM T59328 CCMU48 45483675 IC50 = 23 nM T59328 C9PE3R 45483677 IC50 = 19 nM T59328 CF9SL7 45483685 IC50 = 44 nM T59328 CE7J8I 45483687 IC50 = 30 nM T59328 CULV14 45483689 IC50 = 38 nM T59328 C2V0QA 45483691 IC50 = 40 nM T59328 CFN61Z 45483693 IC50 = 38 nM T59328 CET9K4 45483694 IC50 = 45 nM T59328 CJ1XL4 45483695 IC50 = 21 nM T59328 CO0U2K 45483696 IC50 = 33 nM T59328 CKSM90 45483699 IC50 = 111 nM T59328 C7JH2B 45485483 IC50 = 240 nM T59328 C5QVD7 45485488 IC50 = 180 nM T59328 CN3BQ4 45485489 IC50 = 720 nM T59328 CJ1A3L 45485503 IC50 = 500 nM T59328 CCF08Z 45485522 IC50 = 390 nM T59328 C4HS8N 45485552 IC50 = 770 nM T59328 CB4N0W 46184985 IC50 = 70 nM T59328 C71BUZ 46197015 IC50 < 1 nM T59328 C3HC5D 46197127 IC50 = 16 nM T59328 CZ7W0G 46197128 IC50 = 1.7 nM T59328 CK9Y2G 46197129 IC50 = 30 nM T59328 C5VC7I 46200951 IC50 = 80 nM T59328 C5G7SV 46207008 IC50 = 7820 nM T59328 CA3N9W 46207009 IC50 = 940 nM T59328 C4K9MS 46207010 IC50 = 1720 nM T59328 CAE1M9 46207011 IC50 = 9460 nM T59328 C2F4HI 46207012 IC50 = 11570 nM T59328 C7CID4 46207014 IC50 = 31430 nM T59328 C9CER0 46207015 IC50 > 50000 nM T59328 CPI6S1 46207036 IC50 = 29830 nM T59328 C3F6SM 46207037 IC50 > 50000 nM T59328 C10WUT 46207039 IC50 = 35290 nM T59328 CPXZ65 46207040 IC50 = 22810 nM T59328 C30QNX 46207041 IC50 = 14720 nM T59328 CDN84U 46207042 IC50 = 90 nM T59328 CV1P0R 46207043 IC50 = 17510 nM T59328 C41RBD 46207062 IC50 = 19260 nM T59328 CBQS73 46207441 IC50 = 750 nM T59328 C1WS6M 46207442 IC50 = 1490 nM T59328 CUA97D 46209401 IC50 > 10000 nM T59328 CWN74L 46209503 IC50 = 6900 nM T59328 CKY01V 46209504 IC50 > 10000 nM T59328 CDE1W6 46212905 IC50 = 8 nM T59328 CL41UW 46212970 IC50 = 7 nM T59328 CJR09Y 46212971 IC50 = 0.043 nM T59328 CF57GK 46215462 IC50 = 3900 nM T59328 CY3HW5 46224684 IC50 = 940 nM T59328 C1U7IT 46225595 IC50 = 63 nM T59328 C8YPN0 46225596 IC50 = 350 nM T59328 C34JTS 46225597 EC50 > 10000 nM T59328 CGD73B 46225598 IC50 > 10000 nM T59328 C3E0PU 46225599 IC50 = 4500 nM T59328 CRDY89 46225610 IC50 = 16 nM T59328 C0JMT8 46225611 IC50 = 200 nM T59328 CF0D5J 46225612 IC50 = 46 nM T59328 CFVO38 46225632 IC50 = 2300 nM T59328 CLZ1O6 46225634 IC50 = 805 nM T59328 C07VDX 46225635 IC50 = 670 nM T59328 CT70DX 46225640 IC50 = 32 nM T59328 CJUF68 46225641 IC50 = 44 nM T59328 C6AJ5N 46225647 IC50 = 730 nM T59328 C2WCV1 46225648 IC50 > 10000 nM T59328 CBS96A 46225649 IC50 > 10000 nM T59328 C38BFC 46225657 EC50 = 9400 nM T59328 CD0A6F 46225658 IC50 = 1400 nM T59328 C1B3KS 46225663 IC50 = 430 nM T59328 CU46XI 46225664 IC50 = 260 nM T59328 CO3HS2 46225665 EC50 > 10000 nM T59328 C2UV1S 46225666 EC50 > 10000 nM T59328 CX5B1G 46225667 IC50 = 6200 nM T59328 C2Q9OH 46225668 IC50 = 1400 nM T59328 C16LEO 46225679 IC50 = 2200 nM T59328 CM14FH 46225680 IC50 = 230 nM T59328 CQS96E 46225681 IC50 > 10000 nM T59328 CJIK35 46225682 IC50 = 15 nM T59328 C8S4QA 46225688 IC50 = 250 nM T59328 CYBD14 46229355 IC50 = 1980 nM T59328 C7XEG1 46229356 IC50 = 2240 nM T59328 CO0DJ5 46229377 IC50 = 21710 nM T59328 C5Y1PT 46229378 IC50 = 4150 nM T59328 CE25DB 46229379 IC50 = 4680 nM T59328 CT70VJ 46229380 IC50 = 27350 nM T59328 CT15NR 46229381 IC50 = 960 nM T59328 CG14AQ 46229405 IC50 = 1070 nM T59328 CK7BT5 46229406 IC50 = 7510 nM T59328 CKN40P 46229407 IC50 = 1860 nM T59328 CKL7Z5 46229408 IC50 = 1120 nM T59328 C3IS6A 46229409 IC50 = 9260 nM T59328 CEK82A 46229459 IC50 = 32120 nM T59328 C3N0HQ 46229460 IC50 = 36880 nM T59328 CAO23J 46229461 IC50 > 50000 nM T59328 CJ3FW1 46229462 IC50 > 50000 nM T59328 CI6RL4 46229463 IC50 > 50000 nM T59328 CQ8K2T 46229464 IC50 > 50000 nM T59328 C2SF0M 46229498 IC50 = 670 nM T59328 CY4K7S 46229499 IC50 = 980 nM T59328 C9YBX1 46229500 IC50 = 8540 nM T59328 CF4P3E 46229516 IC50 = 19410 nM T59328 CI1X8G 46229517 IC50 = 120 nM T59328 CH91IA 46229518 IC50 = 3460 nM T59328 CW40RS 46229519 IC50 = 560 nM T59328 CS3OP4 46229535 IC50 = 870 nM T59328 C7UOQ9 46229536 IC50 = 5830 nM T59328 C4MA6T 46229537 IC50 = 18120 nM T59328 CUSX60 46229538 IC50 = 22040 nM T59328 CAKH92 46229539 IC50 = 43210 nM T59328 CLOQ02 46229565 IC50 = 24650 nM T59328 CWD64Q 46229566 IC50 = 31940 nM T59328 CJ4NH6 46229567 IC50 > 50000 nM T59328 C6L0RY 46229767 IC50 = 2.53 nM T59328 CAZ5R0 46229769 IC50 = 87.1 nM T59328 CGMY03 46229773 IC50 = 80 nM T59328 CE12JD 46229813 IC50 = 32.7 nM T59328 CU0RG6 46229815 IC50 > 1000 nM T59328 C31DLC 46229816 IC50 = 32.6 nM T59328 CN2OI5 46229817 IC50 = 106 nM T59328 C5D0OS 46229856 IC50 = 31180 nM T59328 CV96NK 46230527 IC50 = 25.9 nM T59328 C6N7SV 46230529 IC50 = 14.8 nM T59328 C37XZC 46230531 IC50 = 17.7 nM T59328 CYZV41 46231219 IC50 > 8480 nM T59328 C7J5UP 46231220 IC50 = 1688 nM T59328 CC96GZ 46231221 IC50 = 5797 nM T59328 CEOD43 46231624 IC50 = 9120 nM T59328 CXD3E9 46231625 IC50 = 7230 nM T59328 C4J1RQ 46231626 IC50 = 5840 nM T59328 C4XU2C 46231627 IC50 = 4960 nM T59328 CU26ZF 46231684 IC50 = 3110 nM T59328 CA51RN 46231685 IC50 = 1720 nM T59328 CWM8V1 46231686 IC50 = 1010 nM T59328 C2VDX3 46231687 IC50 = 48 nM T59328 CS6I0D 46231742 IC50 = 692 nM T59328 CC0J3D 46231743 IC50 = 1589 nM T59328 CE38ZP 46231744 IC50 = 8710 nM T59328 CTYE12 46231745 IC50 = 6280 nM T59328 C6QG4O 46231746 IC50 = 5330 nM T59328 CE23SX 46231817 IC50 = 3580 nM T59328 CADC90 46231818 IC50 = 2140 nM T59328 C1XV2H 46231819 IC50 = 1270 nM T59328 CLN2B6 46231820 IC50 = 316 nM T59328 CPN4S3 46231883 IC50 = 35 nM T59328 C35LAZ 46231884 IC50 = 464 nM T59328 C5Y3DS 46231885 IC50 = 1350 nM T59328 CYT37A 46232443 IC50 > 50000 nM T59328 C48ZVW 46232555 IC50 > 50000 nM T59328 CS9B1U 46232556 IC50 > 50000 nM T59328 C7ON5A 46233287 IC50 > 10000 nM T59328 CS8P3R 46233390 IC50 = 72 nM T59328 C0QP3Y 46239453 IC50 = 8.59 nM T59328 CZD79U 46831432 IC50 = 12.5 nM T59328 CNWU53 46831433 IC50 = 24.8 nM T59328 C7HK3L 46831434 IC50 = 0.27 nM T59328 CJ9IY2 46831435 IC50 = 0.23 nM T59328 CJ0OF3 46842881 IC50 = 1360 nM T59328 CFP21E 46842882 IC50 = 2170 nM T59328 CN8D3H 46842883 IC50 = 340 nM T59328 CD3TK2 46842884 IC50 = 70 nM T59328 C6UIO0 46842885 IC50 = 130 nM T59328 CGA46B 46842886 IC50 = 3060 nM T59328 CC0I7S 46842887 IC50 = 5190 nM T59328 C9IJ6M 46842888 IC50 = 3870 nM T59328 CBR9Z1 46842916 IC50 = 830 nM T59328 CB2AL1 46842917 IC50 = 4210 nM T59328 CW2BF1 46842918 IC50 = 6270 nM T59328 CIM0F8 46842919 IC50 = 7320 nM T59328 CYTG25 46842920 IC50 = 7780 nM T59328 CUEF65 46842921 IC50 = 11270 nM T59328 CYS9U5 46842922 IC50 = 12260 nM T59328 CDM32Q 46842923 IC50 = 10970 nM T59328 CS3Q7I 46842945 IC50 = 6560 nM T59328 CZ92NO 46842946 IC50 = 7380 nM T59328 C5BGH3 46842947 IC50 = 6850 nM T59328 C9BI7M 46842971 IC50 = 13370 nM T59328 CFR1C6 46845026 IC50 > 300000 nM T59328 CW0P5B 46845702 IC50 = 1060 nM T59328 C7KM0E 46845704 IC50 = 1250 nM T59328 C8ETL6 46854891 IC50 = 82 nM T59328 CKL98B 46854893 IC50 = 452 nM T59328 C0HT9B 46855200 IC50 = 223 nM T59328 C8VX3G 46855360 IC50 = 820 nM T59328 CE3WH9 46865125 IC50 = 4.1 nM T59328 C45LYT 46865445 IC50 = 30.4 nM T59328 CCBE34 46865992 IC50 = 220 nM T59328 C1XEY4 46866615 IC50 = 13.5 nM T59328 CF6K3E 46866616 IC50 = 10.8 nM T59328 CLS29B 46872626 IC50 > 10000 nM T59328 C2MCT8 46879471 IC50 = 867 nM T59328 C6M0JK 46879472 IC50 = 1210 nM T59328 CGV58U 46879473 IC50 > 10000 nM T59328 C8GD2E 46879474 IC50 = 15140 nM T59328 CF4OY7 46881850 IC50 = 58 nM T59328 CEKX49 46881918 IC50 = 58 nM T59328 CMVZ46 46886319 Ki = 31.62 nM T59328 CJR01I 46886321 IC50 = 50 nM T59328 C2O8RZ 46886323 IC50 = 610 nM T59328 CC7MG8 46886325 IC50 = 350 nM T59328 C3T6YO 46886327 IC50 = 1000 nM T59328 CA57MX 46886970 IC50 = 2500 nM T59328 CRGH62 46886971 IC50 = 161600 nM T59328 C68AGR 46886972 IC50 = 27200 nM T59328 CP32GW 46886973 IC50 = 55200 nM T59328 C48JWD 46886974 IC50 = 91700 nM T59328 C7H3MD 46887038 IC50 = 45600 nM T59328 C40NOR 46887039 IC50 = 96400 nM T59328 C7I4SB 46887074 IC50 > 300000 nM T59328 CI5QX2 46887110 IC50 > 300000 nM T59328 C0Q7NG 46887111 IC50 > 300000 nM T59328 CU15AN 46887112 IC50 = 33100 nM T59328 CD90BV 46887113 IC50 > 300000 nM T59328 CH3O9K 46887255 IC50 > 200000 nM T59328 C7NUT3 46887298 IC50 > 200000 nM T59328 CWV65D 46887299 IC50 > 200000 nM T59328 CH5BZ6 46887300 IC50 > 200000 nM T59328 C20UCB 46887348 IC50 > 200000 nM T59328 C0KEG5 46887349 IC50 > 200000 nM T59328 CY59RB 46887397 IC50 = 56100 nM T59328 CL5R0D 46888599 IC50 = 1630 nM T59328 C3IE0X 46888601 IC50 = 980 nM T59328 C1A0XQ 46888603 IC50 = 4400 nM T59328 CB5YQ1 46888635 IC50 = 1920 nM T59328 C6YC4O 46888663 IC50 = 1300 nM T59328 C0AUT8 46888665 IC50 = 2070 nM T59328 CAZT96 46888666 IC50 > 50000 nM T59328 CS4U3P 46888668 IC50 = 2450 nM T59328 CASV10 46888710 IC50 = 1370 nM T59328 CY2TV5 46888712 IC50 = 2750 nM T59328 CX5AL6 46888740 IC50 = 2500 nM T59328 CSWE93 46888742 IC50 = 15120 nM T59328 CW7AR1 46889887 IC50 > 1000 nM T59328 CMNK35 46889911 IC50 > 1000 nM T59328 C0WYM1 46898022 IC50 = 10000 nM T59328 CB92VU 46912443 IC50 > 200000 nM T59328 CU6HC7 46912444 IC50 = 31200 nM T59328 C8A4KU 46912445 IC50 = 1200 nM T59328 CNOS56 46912446 IC50 = 143500 nM T59328 CV38NE 46912546 IC50 = 500 nM T59328 CRI1Q8 46912936 IC50 = 620 nM T59328 C60GAV 46929544 IC50 > 8000 nM T59328 CP34VL 46929748 IC50 > 1000 nM T59328 CJ2E9Q 46929857 IC50 > 25000 nM T59328 C47TGL 46935972 IC50 = 1730 nM T59328 CQVZ79 46935973 IC50 = 2360 nM T59328 CD1N7L 46935974 IC50 = 1840 nM T59328 C7T0ZG 46935975 IC50 = 3850 nM T59328 C12XQO 46936026 IC50 = 2670 nM T59328 C16OAQ 46936027 IC50 = 3080 nM T59328 CBZM62 46936028 IC50 = 1920 nM T59328 C5M0XC 46936029 IC50 = 60 nM T59328 C4H7YB 46936030 IC50 = 190 nM T59328 C19JEL 46936031 IC50 = 370 nM T59328 C6PYR0 46936080 IC50 = 630 nM T59328 CXIN65 46936081 IC50 = 1040 nM T59328 CZ7QW6 46936082 IC50 = 820 nM T59328 CY65UA 46936083 IC50 = 970 nM T59328 CX6A9S 46936084 IC50 = 11240 nM T59328 C4FJA3 46936085 IC50 = 9370 nM T59328 CCUW64 46936126 IC50 = 8950 nM T59328 CS4I3P 46936127 IC50 = 15720 nM T59328 CRKD93 46936128 IC50 = 19640 nM T59328 CR9D8U 46936129 IC50 = 10170 nM T59328 CCHU82 46936130 IC50 = 22360 nM T59328 CE70ZG 46936131 IC50 = 24160 nM T59328 C0IDM5 46936170 IC50 = 17840 nM T59328 C67CSG 46936171 IC50 = 25740 nM T59328 C08QUC 46936172 IC50 = 24370 nM T59328 C9WRB7 46936173 IC50 = 28170 nM T59328 CJ0ZY8 46936174 IC50 = 19830 nM T59328 C60DLE 46936175 IC50 = 21520 nM T59328 CUT3S0 46937464 IC50 = 1.81 nM T59328 C41JQX 46937466 IC50 = 23.02 nM T59328 C2QRW8 46937467 IC50 = 0.57 nM T59328 CONM83 46937468 IC50 = 4.05 nM T59328 C4PZ8J 46937511 IC50 = 0.22 nM T59328 CK5U2C 46937558 IC50 = 0.22 nM T59328 CBZX50 46937560 IC50 = 0.22 nM T59328 C43QHB 46937562 IC50 = 0.22 nM T59328 CBR76Q 46937566 IC50 = 0.22 nM T59328 CPR6O9 47108694 IC50 = 11910 nM T59328 CM24GY 47108695 IC50 = 6740 nM T59328 CF9ZH7 47108713 IC50 = 17810 nM T59328 C4SF5L 47108741 IC50 = 90 nM T59328 CCYJ10 47108773 IC50 = 2080 nM T59328 CJ4T3N 47120995 IC50 = 590 nM T59328 CJS49Y 47232283 IC50 = 3270 nM T59328 CE4SU5 47298428 IC50 > 10000 nM T59328 CCWB05 49788361 IC50 = 720 nM T59328 C0J6HA 49788362 IC50 > 20000 nM T59328 C1OLV6 49788363 IC50 = 1270 nM T59328 CLH4N7 49788364 IC50 = 91 nM T59328 CG0YF3 49788365 IC50 = 3057 nM T59328 COWP56 49788366 IC50 = 20 nM T59328 C93ROW 49788425 IC50 = 46 nM T59328 CM8X1I 49788426 IC50 = 3503 nM T59328 C8XN1P 49788427 IC50 = 9 nM T59328 C3PM9Q 49788428 IC50 = 21 nM T59328 C8AS0L 49788429 IC50 = 89 nM T59328 C31VOW 49788430 IC50 > 20000 nM T59328 C5MZY4 49788490 IC50 = 12 nM T59328 CFLD56 49788491 IC50 = 12 nM T59328 CTQ5M0 49788492 IC50 = 149 nM T59328 CU6Y9D 49788493 IC50 = 4884 nM T59328 C2TY0A 49788560 IC50 > 20000 nM T59328 CE2ST8 49788561 IC50 = 1090 nM T59328 C0EK8U 49788642 IC50 > 20000 nM T59328 CV6O3H 49798025 IC50 = 85 nM T59328 C4FJ0Y 49798860 IC50 = 3880 nM T59328 CBX8W0 49798861 IC50 = 5760 nM T59328 CRLT80 49798983 IC50 = 24150 nM T59328 CL5ZR3 49798984 IC50 = 25470 nM T59328 C26DKM 49798985 IC50 = 15560 nM T59328 CQ80WE 49799021 IC50 = 20610 nM T59328 CX19VP 49799195 IC50 = 8920 nM T59328 CJYK69 49799238 IC50 = 6430 nM T59328 C7NV4K 49799239 IC50 = 7280 nM T59328 C8AWO3 49799240 IC50 = 5270 nM T59328 C37BOI 49799285 IC50 = 17490 nM T59328 CL57XI 49799286 IC50 = 15240 nM T59328 CG3FX1 49799287 IC50 = 21480 nM T59328 C1UPR7 49799323 IC50 = 17310 nM T59328 CO3G7R 49799361 IC50 = 18450 nM T59328 CET2D6 49799362 IC50 = 19320 nM T59328 C05PNX 49799381 IC50 = 16140 nM T59328 CC2WR7 49799382 IC50 = 18350 nM T59328 C7DS9L 49799452 IC50 = 5740 nM T59328 C4B0VH 49799526 IC50 = 10640 nM T59328 CY46VG 49799527 IC50 = 8090 nM T59328 CA26HX 49799528 IC50 = 9830 nM T59328 C69YEO 49799573 IC50 = 10060 nM T59328 CM6HD2 49799574 IC50 = 8150 nM T59328 COD7X8 49799764 IC50 = 3240 nM T59328 C3PNH8 49799765 IC50 = 8110 nM T59328 CO89EH 49799766 IC50 = 10850 nM T59328 C4MYV3 49799767 IC50 = 6820 nM T59328 CK92JP 49799768 IC50 = 1270 nM T59328 CY32VC 49799770 IC50 = 25000 nM T59328 C21GOI 49799777 IC50 = 4120 nM T59328 C7QR3M 49799778 IC50 = 3620 nM T59328 CVEG83 49799781 IC50 = 26740 nM T59328 C6X5MK 49799782 IC50 = 20810 nM T59328 C2GXI7 49799783 IC50 = 24320 nM T59328 C1NI4A 49799785 IC50 = 32000 nM T59328 C3VQ9Z 49799786 IC50 = 14530 nM T59328 CAL42P 49799787 IC50 = 12420 nM T59328 C49XCZ 49799788 IC50 = 13870 nM T59328 CHSF07 49806372 IC50 > 1000 nM T59328 C5ME3S 49806721 IC50 > 50000 nM T59328 C3ZI9B 49840051 IC50 > 10000 nM T59328 CDFE41 49840052 IC50 > 10000 nM T59328 C1XHO0 49840114 IC50 > 10000 nM T59328 CIMT03 49840186 IC50 > 10000 nM T59328 CIX4E3 49840245 IC50 > 10000 nM T59328 CLWN26 49840246 IC50 > 10000 nM T59328 CN89TG 49840317 IC50 > 10000 nM T59328 C0AJ9R 49840318 IC50 > 10000 nM T59328 CF91RS 49843531 IC50 > 10000 nM T59328 CE7D2J 49855568 IC50 = 2.5 nM T59328 CFD9P3 49855569 IC50 = 4.8 nM T59328 C1AU5N 49855758 IC50 = 18 nM T59328 CIFK93 49855759 IC50 = 2.9 nM T59328 CK48OJ 49855760 IC50 = 2.8 nM T59328 CZI3M1 49855761 IC50 = 26 nM T59328 CRPZ58 49855949 IC50 = 49 nM T59328 CTU0K3 49855950 IC50 = 29 nM T59328 CF85NL 49855951 IC50 = 15 nM T59328 CF7YS9 49855952 IC50 = 3.9 nM T59328 CJU38G 49855953 IC50 = 2.2 nM T59328 C9Z8ED 49859891 IC50 = 1000 nM T59328 CB5O0I 49860186 IC50 = 200 nM T59328 C9W6SO 49860190 IC50 = 90 nM T59328 CF4V7Z 49867019 IC50 = 2200 nM T59328 C5RQ7C 50908680 Ki = 500 nM T59328 CD2K4R 50908681 Ki = 400 nM T59328 C6XYT1 50941838 IC50 > 100000 nM T59328 C61DVY 50990961 IC50 = 4900 nM T59328 CV3UP9 50992247 IC50 = 190 nM T59328 CS9G6E 50997096 IC50 > 10000 nM T59328 CM42BY 51000510 Ki = 296000 nM T59328 CAZQ43 51003133 IC50 > 1000 nM T59328 CDU4Q5 51346827 Ki > 1800 nM T59328 C49ZVC 51346878 IC50 = 240 nM T59328 CJ4L1K 51346887 IC50 = 120 nM T59328 CH1TU2 51346888 IC50 = 3 nM T59328 CH1WR3 52914084 IC50 = 149 nM T59328 C13MUQ 52914647 IC50 = 281 nM T59328 CXA03W 52920796 IC50 > 100 nM T59328 CEQN27 52936621 Ki > 1000 nM T59328 CM24LF 52938983 IC50 = 101.4 nM T59328 CAD1N6 52940774 IC50 = 0.03 nM T59328 CU1P2L 52940797 IC50 = 8010 nM T59328 C4R7IM 52941368 IC50 = 253600 nM T59328 C2ZTN3 52941514 IC50 = 2880 nM T59328 CDHJ08 52942235 IC50 = 100000 nM T59328 CG9E4A 52942446 Ki > 1000000 nM T59328 C8SJ2Q 52942862 Ki > 1000000 nM T59328 C7BY6M 52942956 IC50 = 111400 nM T59328 CT8VW3 52943139 IC50 > 10000 nM T59328 C1XEV2 52943394 IC50 = 20500 nM T59328 CA62KU 52944152 IC50 = 160300 nM T59328 CLO46D 52944812 Ki = 3450 nM T59328 CWPC54 52945348 IC50 = 638 nM T59328 CQV34K 52945403 IC50 > 200000 nM T59328 C4NLX7 52945630 IC50 = 54200 nM T59328 CXD6T8 52945845 IC50 = 2800 nM T59328 CQ87LD 52946569 IC50 = 78 nM T59328 C97XZA 52946619 IC50 > 200000 nM T59328 C8QNI5 52946868 IC50 = 8.12 nM T59328 C2WM9K 52947210 IC50 = 5900 nM T59328 CE0X5U 52947574 IC50 > 200000 nM T59328 CD9S4I 52947801 IC50 = 529300 nM T59328 CA6IL3 52947802 IC50 > 200000 nM T59328 CI6GX2 52948511 Ki = 680 nM T59328 C2KAJ4 52948634 IC50 = 53100 nM T59328 CWA74O 52949707 Ki = 590 nM T59328 C0A1GQ 52949915 IC50 = 12800 nM T59328 C6OTY5 53251320 IC50 > 30000 nM T59328 C09SDH 53257410 IC50 > 10000 nM T59328 CX13OD 53316491 IC50 = 150 nM T59328 CJ61BU 53317172 IC50 > 100000 nM T59328 C89QOE 53317173 IC50 = 17 nM T59328 C50BWT 53317174 IC50 = 590 nM T59328 C39KUD 53317175 IC50 = 38 nM T59328 C1NLD5 53317828 IC50 = 4100 nM T59328 CE8OY2 53317913 IC50 > 100 nM T59328 CBHT02 53318117 IC50 = 950 nM T59328 CX1V9L 53318118 IC50 = 670 nM T59328 C90MNQ 53318457 IC50 = 1100 nM T59328 C2X8OF 53318458 IC50 = 18 nM T59328 CK59QY 53318459 IC50 = 270 nM T59328 CZS8K4 53319042 Ki > 1800 nM T59328 C3MUN7 53319130 IC50 = 2200 nM T59328 C1PMT2 53319131 IC50 = 55600 nM T59328 CRBE56 53319790 IC50 = 34 nM T59328 CSC61X 53320059 IC50 = 114 nM T59328 CUD21V 53320263 Ki > 1800 nM T59328 C4QU3S 53320463 IC50 = 6900 nM T59328 CX65KS 53321087 IC50 = 10000 nM T59328 C3G2WX 53321754 IC50 = 28000 nM T59328 CX7S8I 53322057 IC50 > 1000 nM T59328 CSY76U 53322058 IC50 = 210 nM T59328 C7Y3ZR 53322413 IC50 = 640 nM T59328 CR12OB 53322414 IC50 = 156 nM T59328 CR4K7J 53322690 IC50 = 65 nM T59328 CESA85 53323614 Ki > 1800 nM T59328 CT1BN7 53324027 IC50 = 47000 nM T59328 C43BZJ 53324200 IC50 = 20000 nM T59328 CI6A9B 53324357 IC50 = 1300 nM T59328 CB80KQ 53324440 IC50 = 12800 nM T59328 CGL6Y7 53324441 IC50 = 45200 nM T59328 CG18XC 53325046 IC50 = 1200 nM T59328 CD91UQ 53325047 IC50 = 22000 nM T59328 C5C1UW 53325048 IC50 = 68 nM T59328 CRT07X 53325049 IC50 = 28 nM T59328 C69AUF 53325050 IC50 = 11 nM T59328 CN1X9I 53325551 IC50 = 19 nM T59328 C36OQR 53325588 IC50 > 1000 nM T59328 CNX76J 53325743 IC50 = 20800 nM T59328 C07PMQ 53326342 IC50 = 4130 nM T59328 CD86WI 53328229 IC50 = 4 nM T59328 C5ETO8 53328965 IC50 = 3 nM T59328 CCZG21 53328969 IC50 = 1600 nM T59328 CJ2Y5P 53330551 IC50 = 13 nM T59328 CNPM14 53341082 IC50 = 3.3 nM T59328 C0SWH5 53348216 IC50 > 40000 nM T59328 C8ZRE3 53356518 IC50 > 16670 nM T59328 CM7P3W 53357328 IC50 > 50000 nM T59328 C4PO3Z 53357348 IC50 = 1929 nM T59328 CXW05L 53357349 IC50 = 12070 nM T59328 CBK9Q6 53357848 IC50 > 10000 nM T59328 C8NA4L 53384644 IC50 > 30000 nM T59328 CVG90B 53389651 IC50 > 10000 nM T59328 CA50GN 53466759 IC50 < 7 nM T59328 CJ1NB9 53484041 IC50 = 940 nM T59328 CREZ21 53484042 IC50 = 120 nM T59328 C0HN6L 53484043 IC50 = 190 nM T59328 C8D9XG 53736592 IC50 > 10000 nM T59328 C9MBJ6 53759588 IC50 = 4.7 nM T59328 CH53KW 54576742 IC50 = 350 nM T59328 CK1EM6 54580365 IC50 > 10000 nM T59328 C4SN3X 54580366 IC50 > 10000 nM T59328 CQ9I1X 54580996 IC50 = 67 nM T59328 C1HZ4Y 54581368 IC50 > 10000 nM T59328 CA6H2U 54581369 IC50 > 10000 nM T59328 C5P9BQ 54581370 IC50 > 10000 nM T59328 CW7NH3 54582387 IC50 > 10000 nM T59328 C7R4UG 54582388 IC50 > 10000 nM T59328 C9SZ2I 54582389 IC50 > 10000 nM T59328 CL40KE 54583375 IC50 > 10000 nM T59328 C2MFX7 54585296 IC50 > 10000 nM T59328 CY4RH6 54586238 IC50 > 10000 nM T59328 C8QA0M 54586239 IC50 > 10000 nM T59328 C6RX7G 54586507 IC50 = 95 nM T59328 CL1I5C 54587267 IC50 > 10000 nM T59328 C0JMY7 54673975 IC50 = 82900 nM T59328 CUT84L 54678831 IC50 > 100000 nM T59328 CZH60Y 54708982 IC50 = 76400 nM T59328 CUZH35 54754343 IC50 = 390 nM T59328 C1XS2J 54760383 IC50 = 4 nM T59328 C75YDA 54768720 IC50 = 2080 nM T59328 C65TFD 54768721 IC50 = 10950 nM T59328 C1WVC6 54768722 IC50 = 19120 nM T59328 C05SPN 54768723 IC50 = 20480 nM T59328 CRL5O0 54768724 IC50 = 26560 nM T59328 CBN0C3 54768725 IC50 = 17390 nM T59328 CR98HI 54768726 IC50 = 14830 nM T59328 C7B8XU 54768951 IC50 = 1570 nM T59328 CT1P3J 54768952 IC50 = 5110 nM T59328 CMN8T0 54768953 IC50 = 700 nM T59328 CZEC06 54768954 IC50 = 2380 nM T59328 C21KRM 54768955 IC50 = 12240 nM T59328 CJ0Q4M 54768956 IC50 = 8660 nM T59328 CY7B5N 54768957 IC50 = 590 nM T59328 CJAN-67 54768958 IC50 = 9780 nM T59328 CE0O9W 54769185 IC50 = 2170 nM T59328 C8LI9H 54769186 IC50 = 7830 nM T59328 CZE0I1 54769187 IC50 = 410 nM T59328 CE8WK1 54772084 IC50 = 22360 nM T59328 CPMZ93 54772085 IC50 = 23270 nM T59328 CKA7U0 54772086 IC50 = 26000 nM T59328 CC4FN9 54772087 IC50 = 33000 nM T59328 CU8YW6 56325569 IC50 = 45000 nM T59328 CQ17GA 56640518 IC50 = 34.8 nM T59328 CG20VK 56640520 IC50 = 6.8 nM T59328 CZ9C8M 56640588 IC50 = 14.7 nM T59328 CH0D7P 56640590 IC50 = 17.6 nM T59328 CN9QD7 56643097 IC50 > 10000 nM T59328 CK2F5X 56649610 IC50 = 66100 nM T59328 CTF90E 56649640 IC50 = 6.6 nM T59328 CU76CR 56649641 IC50 = 3.8 nM T59328 C1LQT6 56649642 IC50 = 3.3 nM T59328 CT6G3J 56649645 IC50 > 100000 nM T59328 C5D4EP 56659276 IC50 = 60 nM T59328 CPZ62X 56659321 IC50 = 6020 nM T59328 C9XCI1 56659322 IC50 = 1020 nM T59328 CR6VD1 56659589 IC50 = 251.19 nM T59328 C2PYI1 56659875 IC50 = 11290 nM T59328 CT5NK2 56659876 IC50 = 18350 nM T59328 C2MW9D 56659883 IC50 = 21280 nM T59328 CX28ME 56660000 IC50 > 10000 nM T59328 CYZ6C5 56661789 IC50 = 8630 nM T59328 CD0UZ8 56662784 IC50 = 3610 nM T59328 CNE6P1 56662786 IC50 = 2810 nM T59328 CD67RU 56663333 IC50 = 13730 nM T59328 CCR3V9 56663334 IC50 = 24150 nM T59328 C6QY0W 56665233 IC50 = 5560 nM T59328 C7NF0U 56666765 IC50 = 2940 nM T59328 C9LPB6 56666766 IC50 = 21840 nM T59328 C4S9ID 56666767 IC50 = 32850 nM T59328 CT3BC2 56669670 IC50 = 8800 nM T59328 C4L2QB 56670196 IC50 = 3430 nM T59328 CIPW74 56670197 IC50 = 1510 nM T59328 CSNH68 56670198 IC50 = 15920 nM T59328 C97LHS 56670199 IC50 = 17260 nM T59328 C6W7BR 56670200 IC50 = 38520 nM T59328 CK2B0C 56672168 IC50 = 6310 nM T59328 CS45AF 56673177 IC50 = 3490 nM T59328 CRXF95 56673721 IC50 = 5930 nM T59328 CG9N7C 56673722 IC50 = 6410 nM T59328 CFAT97 56673723 IC50 = 26200 nM T59328 CT85LD 56676436 IC50 = 1210 nM T59328 CL2DT3 56676437 IC50 = 4280 nM T59328 CMO70N 56676438 IC50 = 7220 nM T59328 CXP5G4 56677027 IC50 = 14530 nM T59328 CE40HN 56678885 IC50 = 8430 nM T59328 C6ME8I 56680356 IC50 = 2170 nM T59328 CNLI27 56680357 IC50 = 8280 nM T59328 CN28KJ 56680358 IC50 = 9590 nM T59328 CYT34H 56682199 IC50 = 5350 nM T59328 C21SXU 56682201 IC50 = 7660 nM T59328 CV3QB9 56683074 IC50 = 7710 nM T59328 CX2MU1 56683151 IC50 = 5160 nM T59328 CG6JP0 56683152 IC50 = 6630 nM T59328 CC2E5V 56683153 IC50 = 3450 nM T59328 COK71Z 56683687 IC50 = 5170 nM T59328 CQ8Z1X 56683695 IC50 = 24680 nM T59328 C5GM0Z 56683696 IC50 = 26170 nM T59328 CNL0A1 56683697 IC50 = 18720 nM T59328 CP7M1A 56683698 IC50 = 24330 nM T59328 C12XMC 56735038 IC50 = 38320 nM T59328 CR50TJ 56835147 IC50 > 10000 nM T59328 CI5ZJ7 56835161 IC50 = 190 nM T59328 CVA8U4 56837416 IC50 = 870 nM T59328 C3QD4K 56839586 IC50 = 16.6 nM T59328 CLSN24 56839587 IC50 = 5.54 nM T59328 CW06VF 56839588 IC50 = 24 nM T59328 CRYP21 56839589 IC50 = 5.93 nM T59328 CJRC62 56849701 IC50 = 34 nM T59328 CG5O8V 56933480 IC50 = 47900 nM T59328 C4P2LY 56934730 IC50 = 63 nM T59328 C63NMS 56934846 IC50 = 33 nM T59328 CP9OF7 56934847 IC50 = 27 nM T59328 CP97GH 56934848 IC50 = 29 nM T59328 CGLB90 56934849 IC50 = 14 nM T59328 C8KV0I 56934851 IC50 = 62 nM T59328 CFK7L9 56934853 IC50 = 450 nM T59328 CXN79H 56934855 IC50 = 4608 nM T59328 C42EHX 56934976 IC50 = 8 nM T59328 CXC51G 56934978 IC50 = 17 nM T59328 COM4F5 56934980 IC50 = 9 nM T59328 C54DNK 56934982 IC50 = 95 nM T59328 C1N4LK 56934984 IC50 = 26 nM T59328 C8O0IR 56934986 IC50 = 52 nM T59328 CBO20L 56934988 IC50 = 45 nM T59328 C2XED0 56935104 IC50 = 4 nM T59328 C8JZC2 56935107 IC50 = 1008 nM T59328 CGV1M9 56935337 IC50 = 93300 nM T59328 CAW57M 56935338 IC50 > 100000 nM T59328 C76EOA 56935464 IC50 > 100000 nM T59328 CO62XN 56935468 IC50 > 100000 nM T59328 CQ2U4F 56949987 IC50 = 37 nM T59328 C86USY 56950114 IC50 = 61 nM T59328 CCTI03 56950115 IC50 = 48 nM T59328 C5K3PV 56950116 IC50 = 65 nM T59328 C7U9SL 56951304 IC50 > 50000 nM T59328 C0GQ9I 56951305 IC50 = 112100 nM T59328 C5YT6A 56951306 IC50 = 12620 nM T59328 CB03EH 56951307 IC50 > 200000 nM T59328 CRJ6H8 56953639 IC50 > 10000 nM T59328 C3D6YR 56953640 IC50 > 10000 nM T59328 CZ9F6B 56953642 IC50 > 10000 nM T59328 CTDR35 56953644 IC50 > 10000 nM T59328 CYF6D8 56953645 IC50 = 9800 nM T59328 CR20WU 56953646 IC50 = 9150 nM T59328 C86GAQ 56953648 IC50 > 10000 nM T59328 CMRB39 56953766 IC50 > 10000 nM T59328 CNG63B 56953767 IC50 > 10000 nM T59328 C1OC9P 56953892 IC50 > 10000 nM T59328 CF5AV8 56953893 IC50 > 10000 nM T59328 CBHG03 56953894 IC50 > 10000 nM T59328 CB5I7C 56953895 IC50 = 7050 nM T59328 C1NIS7 56954003 IC50 = 800 nM T59328 CEKO58 56954004 IC50 = 4800 nM T59328 C7FP1R 56954005 IC50 = 6150 nM T59328 C0PY2A 56954006 IC50 = 1000 nM T59328 CU1QF7 56954007 IC50 = 1000 nM T59328 CG9X1J 56954008 IC50 = 6400 nM T59328 CM9Z4I 56954009 IC50 = 4000 nM T59328 CX1U4G 56954130 IC50 = 900 nM T59328 CG1VI6 56954131 IC50 = 900 nM T59328 CLR6J2 56954132 IC50 = 7600 nM T59328 C9OZ7N 56954133 IC50 = 5800 nM T59328 CLJC74 56954134 IC50 = 900 nM T59328 CEWB79 56954135 IC50 = 7200 nM T59328 CY2GE9 56954136 IC50 = 5000 nM T59328 C5ATX6 56954232 IC50 > 10000 nM T59328 CU3T6F 56954234 IC50 > 10000 nM T59328 CMWK36 56954235 IC50 = 9900 nM T59328 CM9O5W 56954236 IC50 > 10000 nM T59328 C35JTA 56954323 IC50 = 9450 nM T59328 CI5MT0 56954324 IC50 > 10000 nM T59328 C06IDB 56954325 IC50 > 10000 nM T59328 CMT80I 56954326 IC50 > 10000 nM T59328 CE68LB 56954327 IC50 > 10000 nM T59328 CA43UF 56954328 IC50 > 10000 nM T59328 CC85JQ 56954429 IC50 = 9100 nM T59328 CP58NG 56954518 IC50 > 10000 nM T59328 C7K1CZ 56954519 IC50 > 10000 nM T59328 CH1X3R 56954520 IC50 > 10000 nM T59328 CMS50D 56954621 IC50 > 10000 nM T59328 C30ALB 56954622 IC50 > 10000 nM T59328 CZN89G 56954623 IC50 > 10000 nM T59328 CI7U1E 56954736 IC50 > 10000 nM T59328 C18BFU 56954737 IC50 > 10000 nM T59328 CO7D3X 56954739 IC50 > 10000 nM T59328 CRZ0M5 56954836 IC50 = 7050 nM T59328 C04JZF 56954837 IC50 = 800 nM T59328 CH98NL 56954839 IC50 = 6150 nM T59328 CN06PL 56954840 IC50 = 1000 nM T59328 CH0SG3 56954841 IC50 = 1000 nM T59328 C3MYG6 56954954 IC50 = 6400 nM T59328 C6WAD7 56954955 IC50 = 4000 nM T59328 CZ82IH 56954956 IC50 = 900 nM T59328 CSBQ86 56954957 IC50 = 900 nM T59328 CIM60L 56954958 IC50 = 7600 nM T59328 C1LC4G 56955061 IC50 = 900 nM T59328 C4OY1T 56955062 IC50 = 7200 nM T59328 CSJ6L7 56955063 IC50 = 5000 nM T59328 C1GA2O 56955275 IC50 > 10000 nM T59328 CT1KX9 56955277 IC50 > 10000 nM T59328 CAK91L 56955954 IC50 = 739 nM T59328 CJ47MX 56963907 IC50 > 10000 nM T59328 C9L6FD 56963908 IC50 > 10000 nM T59328 CE50IB 56963909 IC50 > 10000 nM T59328 CIX32Y 56965877 IC50 = 2820 nM T59328 COXM57 56970372 IC50 = 1510 nM T59328 CPHX64 57325478 IC50 > 50000 nM T59328 CQ9BW4 57325479 IC50 > 50000 nM T59328 CJ0A7O 57336240 IC50 = 7 nM T59328 CW2G7E 57341100 IC50 = 1.47 nM T59328 CF0RI1 57341101 IC50 = 3.52 nM T59328 CE7ID2 57341102 IC50 = 6.95 nM T59328 C5U4EK 57341103 IC50 = 929 nM T59328 CJ14YA 57341104 IC50 = 0.43 nM T59328 C7VX2L 57341295 IC50 = 0.41 nM T59328 C5UC3L 57341296 IC50 = 4.41 nM T59328 CJY51G 57341297 IC50 = 8.81 nM T59328 CTA57G 57341298 IC50 = 1.95 nM T59328 CW7H2P 57341299 IC50 > 1000 nM T59328 CQ0D5S 57341488 IC50 = 0.38 nM T59328 C2L0VD 57341489 IC50 = 0.58 nM T59328 C7WU1S 57341490 IC50 = 0.3 nM T59328 CX01VB 57341491 IC50 = 0.8 nM T59328 C8C4DZ 57341660 IC50 = 0.29 nM T59328 CQR64D 57341661 IC50 = 1.41 nM T59328 CS4YT2 57341662 IC50 = 1.52 nM T59328 CVG52R 57341663 IC50 = 1.67 nM T59328 CFDQ12 57341838 IC50 > 1000 nM T59328 CT53HQ 57341839 IC50 > 1000 nM T59328 CBJW71 57343703 IC50 = 1.16 nM T59328 C34OGM 57343704 IC50 = 4.99 nM T59328 CB0DY1 57343705 IC50 = 29.5 nM T59328 CW7B3X 57343706 IC50 = 16.4 nM T59328 CVD3B0 57381322 IC50 = 65 nM T59328 C2JD7G 57381323 IC50 = 31 nM T59328 CD65MT 57381324 IC50 = 15 nM T59328 C4YFJ5 57384105 IC50 > 200000 nM T59328 CV9RW5 57384106 IC50 > 200000 nM T59328 C8O4DU 57390197 IC50 = 473 nM T59328 C0E5UQ 57390198 IC50 = 108 nM T59328 CLB4Q9 57390199 IC50 = 129 nM T59328 C04YLM 57390200 IC50 > 10000 nM T59328 CT6GK0 57390220 IC50 > 100000 nM T59328 COC5Y3 57390776 IC50 = 9 nM T59328 C20OVM 57390777 IC50 = 24 nM T59328 CNB25Q 57390936 IC50 = 15680 nM T59328 CR4T2Y 57391283 IC50 > 200000 nM T59328 C80RNH 57391987 IC50 = 1671 nM T59328 C8U9EO 57391988 IC50 = 627 nM T59328 CXL95C 57392008 IC50 > 100000 nM T59328 CK04XQ 57392009 IC50 > 100000 nM T59328 CBL74E 57392425 IC50 > 200000 nM T59328 CHS82P 57392588 IC50 = 7 nM T59328 CZBJ71 57392589 IC50 = 79 nM T59328 CH12GK 57392590 IC50 = 74 nM T59328 CY2XK0 57392591 IC50 = 94 nM T59328 CC2AF6 57392917 IC50 = 25360 nM T59328 CTB8R9 57394107 IC50 = 821 nM T59328 CLY6T8 57394393 IC50 > 30000 nM T59328 CH1U8Y 57394394 IC50 = 2640 nM T59328 CE1A9V 57394653 IC50 = 1.4 nM T59328 CNV76Z 57394656 IC50 = 3.35 nM T59328 CG18LI 57394786 IC50 > 200000 nM T59328 CEDP89 57394787 IC50 > 200000 nM T59328 CP6W4C 57394879 IC50 = 166400 nM T59328 CVR13L 57394880 IC50 = 99900 nM T59328 C8W6IG 57395117 IC50 > 30000 nM T59328 CJC5N7 57395350 IC50 = 18.5 nM T59328 CN7S2K 57395407 IC50 = 1640 nM T59328 C9NA7R 57395419 IC50 = 1870 nM T59328 C9CO0F 57395424 IC50 > 10000 nM T59328 CA4Q3Y 57395925 IC50 = 112700 nM T59328 CM18WP 57396070 IC50 = 86 nM T59328 C2HT3R 57396157 IC50 > 30000 nM T59328 CVA2E1 57396158 IC50 = 21560 nM T59328 CGE48O 57396218 IC50 = 27050 nM T59328 CX1S8R 57396219 IC50 = 28660 nM T59328 CUGP85 57396545 IC50 > 200000 nM T59328 CBUP96 57396646 IC50 = 113300 nM T59328 CI3JB2 57396795 IC50 > 100000 nM T59328 CA02UC 57397177 IC50 = 43.7 nM T59328 CSKH73 57397251 IC50 = 3220 nM T59328 CSAZ51 57397252 IC50 = 11220 nM T59328 C0GSP4 57397265 IC50 = 4410 nM T59328 C6NC2K 57397269 IC50 = 370 nM T59328 CWX47O 57397293 IC50 > 100000 nM T59328 C87OHQ 57397677 IC50 > 10000 nM T59328 CO24DL 57397871 IC50 = 22 nM T59328 C5D1MK 57397872 IC50 = 30 nM T59328 CI6UJ0 57397973 IC50 = 29070 nM T59328 C58KTL 57397974 IC50 = 18150 nM T59328 C18HFC 57397975 IC50 = 15020 nM T59328 CNLS72 57398015 IC50 = 19830 nM T59328 CXJ68F 57398331 IC50 > 200000 nM T59328 C14ANY 57398417 IC50 = 69200 nM T59328 CGV35E 57398558 IC50 > 100000 nM T59328 C73MUW 57398687 IC50 = 422 nM T59328 C9RA2M 57398688 IC50 = 342 nM T59328 C8EB1H 57398880 IC50 = 18.7 nM T59328 CNA4C0 57398939 IC50 = 3130 nM T59328 C7ZI0C 57398942 IC50 = 3540 nM T59328 CG9E5X 57399346 IC50 = 523 nM T59328 C9U2ZS 57399744 IC50 = 12 nM T59328 C2GJQ6 57399859 IC50 > 30000 nM T59328 CDF35C 57400360 IC50 = 9021 nM T59328 C8ZYQ6 57400361 IC50 = 9284 nM T59328 CO34ZJ 57400426 IC50 = 55 nM T59328 CH1A8D 57400659 IC50 = 13880 nM T59328 CC3U6B 57400808 IC50 > 40000 nM T59328 CQ5MB9 57401285 IC50 = 650 nM T59328 CMP96A 57401286 IC50 = 98 nM T59328 C0WFY5 57401428 IC50 > 30000 nM T59328 CTX6K2 57401429 IC50 > 30000 nM T59328 CV1K0D 57401637 IC50 > 30000 nM T59328 C9MAH3 57402380 IC50 = 10.8 nM T59328 C9ZKD5 57402437 IC50 = 5670 nM T59328 CKVJ46 57402440 IC50 = 1204 nM T59328 CP2UN4 57402469 IC50 = 29500 nM T59328 CD0W6U 57402866 IC50 = 721 nM T59328 C1B7RI 57403128 IC50 = 1190 nM T59328 CKFJ31 57403923 IC50 = 623 nM T59328 CZSM95 57412684 IC50 > 10000 nM T59328 CT7M3G 57413593 IC50 = 5.5 nM T59328 CM9OF3 57413596 IC50 = 7 nM T59328 C1RS3Y 57415414 IC50 = 7.8 nM T59328 C80BOQ 57415415 IC50 = 510 nM T59328 CSV93M 57415416 IC50 = 960 nM T59328 C3H6UJ 57415417 IC50 = 2300 nM T59328 CW5IS7 57415418 IC50 = 890 nM T59328 C1DS4B 57415535 IC50 = 21 nM T59328 C0W8LA 57415536 IC50 = 2.8 nM T59328 CRB83E 57415537 IC50 = 36 nM T59328 CN53XW 57428969 IC50 = 283.1 nM T59328 CI5U3G 57496699 IC50 = 11 nM T59328 CZ35GD 57496700 IC50 = 33 nM T59328 C4T7PW 57523998 IC50 > 10000 nM T59328 C1Q7LS 57523999 IC50 = 82 nM T59328 CPS79I 57524088 IC50 = 2350 nM T59328 C0CJ8Z 57524184 IC50 = 3315 nM T59328 C8ICV2 57524400 IC50 = 99 nM T59328 CL72NQ 57524403 IC50 = 165 nM T59328 CAU0K1 57524478 IC50 = 188 nM T59328 CWVJ06 57597166 IC50 = 15 nM T59328 CVS51B 57597223 IC50 = 53 nM T59328 C0QUZ4 57597316 IC50 = 47 nM T59328 CD0M7X 57597387 IC50 = 18 nM T59328 CVK0G4 58056356 IC50 > 50000 nM T59328 C4V7FY 58191950 IC50 = 1300 nM T59328 CPCA29 58191961 IC50 = 1200 nM T59328 C7HF1L 58191965 IC50 = 78 nM T59328 C8LWY9 58191997 IC50 = 33 nM T59328 C3VI7D 58229394 IC50 = 650 nM T59328 CNXU29 58229412 IC50 = 1128 nM T59328 C52OMW 58229434 IC50 = 592 nM T59328 C6BPR2 58985201 IC50 > 50000 nM T59328 C40EXM 59151065 IC50 < 1 nM T59328 C1SI3L 59174579 IC50 = 737 nM T59328 CXN56R 59174683 IC50 = 500 nM T59328 CT3EW2 59292007 IC50 > 1000 nM T59328 C2FYK8 59322489 IC50 = 82 nM T59328 C6NCJ4 59322491 IC50 = 7893 nM T59328 CS35WB 59322547 IC50 = 352 nM T59328 CN6PF7 59322583 IC50 = 589 nM T59328 CH5SO4 59322599 IC50 > 10000 nM T59328 C3KTW7 59322608 IC50 = 434 nM T59328 CGH6T7 59322651 IC50 = 179 nM T59328 CX2WH5 59322657 IC50 = 64 nM T59328 C9AEM1 59322682 IC50 = 218 nM T59328 C19QYP 59322697 IC50 = 3.9 nM T59328 C0YG3I 59322699 IC50 = 9 nM T59328 C9GWZ0 59322716 IC50 = 258 nM T59328 C52WSD 59322732 IC50 = 0.214 nM T59328 C67WFH 59322756 IC50 = 159 nM T59328 C7PE3G 59453176 IC50 = 6.9 nM T59328 CHC3W6 59484610 IC50 = 38 nM T59328 C1B3NR 59484612 IC50 = 110 nM T59328 CX0KC2 59484694 IC50 = 75 nM T59328 CXJ63M 59603829 IC50 = 28000 nM T59328 CQEU96 59603842 IC50 = 340 nM T59328 CXG78H 60020799 IC50 = 2991 nM T59328 C1MR8Q 60097495 IC50 > 1000 nM T59328 CSZA16 60155724 IC50 = 410 nM T59328 CK8EN9 60166357 IC50 = 59 nM T59328 CU79HD 60202383 IC50 = 2 nM T59328 C9ZCT2 62705065 IC50 > 1000 nM T59328 CUBL90 66545750 IC50 = 1620 nM T59328 CY5KC6 66550688 IC50 = 230 nM T59328 C4K2VC 66550892 IC50 = 1350 nM T59328 CK6WO0 66552478 IC50 < 10000 nM T59328 C10AMI 66553589 IC50 > 10000 nM T59328 C7CW0V 66554568 IC50 = 104.7 nM T59328 CPT48Z 66554916 IC50 = 167.3 nM T59328 C9ABY5 66555108 IC50 = 32.2 nM T59328 CID49H 66555110 IC50 = 5.8 nM T59328 C1FZ9G 66555254 IC50 = 100.1 nM T59328 CA2MK9 66555427 IC50 = 72.2 nM T59328 CB5RC1 66555609 IC50 > 1000 nM T59328 CE0U3J 66555781 IC50 = 1.8 nM T59328 CY6LN5 66555942 IC50 > 1000 nM T59328 C8N5KT 66555946 IC50 = 195.8 nM T59328 CQ61CB 66556107 IC50 = 102.2 nM T59328 CH35UQ 66556108 IC50 = 115.1 nM T59328 CXI2E5 66556610 IC50 = 121.1 nM T59328 CF5A3X 66556780 IC50 = 8.1 nM T59328 CRDU73 66556783 IC50 = 134.9 nM T59328 CWSJ26 66556966 IC50 = 560.4 nM T59328 C9QF6B 66559005 IC50 = 27 nM T59328 C1HSE0 67035086 IC50 = 2300 nM T59328 CWI6K5 67035106 IC50 > 10000 nM T59328 C38RGB 67035556 IC50 > 10000 nM T59328 CV3HW2 67035568 IC50 > 10000 nM T59328 CD14OC 67071561 IC50 = 3081 nM T59328 CEKN37 67073846 IC50 = 178 nM T59328 CR8L3N 67128637 IC50 = 3150 nM T59328 C7B9GO 67128667 IC50 = 8870 nM T59328 CWT14V 67137892 IC50 = 63.4 nM T59328 CV63UL 67240318 IC50 > 10000 nM T59328 C5SYC3 67304928 IC50 = 170 nM T59328 CR1ZL0 67346310 IC50 = 25 nM T59328 CCAD76 68196023 IC50 = 41 nM T59328 C8I7GC 68293638 IC50 > 10000 nM T59328 CD56XK 68293660 IC50 > 10000 nM T59328 CU57RD 68304261 IC50 > 25000 nM T59328 CI0A4N 68304989 IC50 = 400 nM T59328 C76TLN 68305106 IC50 = 630 nM T59328 C1FD5A 68342470 IC50 = 3100 nM T59328 C7WP9L 68342530 IC50 = 1700 nM T59328 C3JE5H 68356029 IC50 = 285 nM T59328 CNC27X 68594933 IC50 = 203 nM T59328 C57ENP 68629464 IC50 = 3 nM T59328 CG7KR4 68669354 IC50 = 9.8 nM T59328 CZB4E9 68672618 Ki = 22 nM T59328 CBIL54 68678227 IC50 > 10000 nM T59328 CAIO65 68796885 IC50 = 112 nM T59328 C5DGR9 69036886 IC50 = 10000 nM T59328 CW0E7O 69104616 IC50 = 257 nM T59328 CVN97F 69714349 IC50 = 109 nM T59328 CE5U7A 69956412 IC50 = 130016.96 nM T59328 C73ZTD 70023804 IC50 > 100000 nM T59328 C7IZW8 70681324 IC50 = 11 nM T59328 CK2G8E 70681325 IC50 = 0.49 nM T59328 CXRF43 70681934 IC50 = 2340 nM T59328 CLK09M 70681935 IC50 = 1800 nM T59328 CX5VN1 70681936 IC50 = 6170 nM T59328 C1ALW8 70682361 IC50 = 30000 nM T59328 CXW0E5 70682363 IC50 = 4500 nM T59328 CT5R9G 70682364 IC50 = 65000 nM T59328 CGM71F 70683719 IC50 = 0.29 nM T59328 CE3VQ2 70683720 IC50 = 0.68 nM T59328 C6USH3 70683721 IC50 = 37.5 nM T59328 CS30XY 70684051 IC50 = 1410 nM T59328 C9OT4C 70684052 IC50 = 1410 nM T59328 C5FYX7 70684449 IC50 = 1400 nM T59328 CJ83GE 70684450 IC50 = 6800 nM T59328 CNI19U 70684611 IC50 = 790 nM T59328 CDT70C 70684612 IC50 = 1290 nM T59328 C5DN2W 70684613 IC50 = 630 nM T59328 C9J0BO 70684614 IC50 = 216 nM T59328 CK83NM 70685870 IC50 = 17.4 nM T59328 C0JV2Y 70685871 IC50 = 2.21 nM T59328 C4M2OY 70686190 IC50 = 2220 nM T59328 CQE6H8 70686191 IC50 = 3530 nM T59328 CLT47X 70686585 IC50 = 230 nM T59328 CEV43U 70686586 IC50 = 140 nM T59328 CR5NW7 70686587 IC50 = 3000 nM T59328 C7L5MA 70686588 IC50 = 7800 nM T59328 CVH29P 70686589 IC50 = 120 nM T59328 C82FIP 70686752 IC50 = 700 nM T59328 CVP42W 70686767 IC50 = 1630 nM T59328 C7EM5X 70686945 IC50 = 120 nM T59328 CKCU42 70687611 IC50 > 10000 nM T59328 CE8LV1 70688705 IC50 = 61 nM T59328 C0QX3Y 70688829 IC50 = 510 nM T59328 CYP97H 70688851 IC50 = 570 nM T59328 C47IRO 70688852 IC50 = 1140 nM T59328 CDI67X 70689230 IC50 = 419 nM T59328 C24TEK 70690021 IC50 = 0.27 nM T59328 CC3D2S 70690022 IC50 = 1.46 nM T59328 C8KS2X 70690332 IC50 = 4200 nM T59328 C29RZD 70690333 IC50 = 2250 nM T59328 CM9C6X 70690334 IC50 = 900 nM T59328 C57QVT 70690769 IC50 = 78 nM T59328 C1OLS7 70690770 IC50 = 5800 nM T59328 CCT2Z7 70690771 IC50 = 75000 nM T59328 CT6CN0 70690772 IC50 = 570 nM T59328 CIJ57N 70690773 IC50 = 79000 nM T59328 CEQP73 70690935 IC50 = 98 nM T59328 CF30HQ 70692178 IC50 = 2.02 nM T59328 CXG2I4 70692907 IC50 = 380 nM T59328 CBS26Q 70692909 IC50 = 67 nM T59328 CH85TX 70692910 IC50 = 7200 nM T59328 CSOT12 70693058 IC50 > 10000 nM T59328 CS6NW3 70693059 IC50 > 10000 nM T59328 CR67GN 70693078 IC50 = 3680 nM T59328 CUT1L7 70693079 IC50 = 920 nM T59328 C1SF0B 70693242 IC50 = 5 nM T59328 CQ5W6D 70693519 IC50 = 6 nM T59328 C4N6ZM 70693874 IC50 > 10000 nM T59328 CS64HU 70694243 IC50 = 0.18 nM T59328 C68TLE 70694244 IC50 = 0.51 nM T59328 CP4V0G 70694245 IC50 = 50.7 nM T59328 CO1MU8 70694542 IC50 = 1100 nM T59328 C9D4UF 70694543 IC50 = 1120 nM T59328 CA0CP1 70694544 IC50 = 5160 nM T59328 CWM62Q 70694846 Ki > 10000 nM T59328 CHF7G6 70694948 IC50 = 3700 nM T59328 CI52UN 70695327 IC50 = 7 nM T59328 C6HI8Q 70696598 IC50 = 3310 nM T59328 CBCF23 70696599 IC50 = 1560 nM T59328 CW8A5I 70697001 IC50 = 380 nM T59328 C59NUJ 70697002 IC50 = 990 nM T59328 CWDR98 70697003 IC50 = 99 nM T59328 C3JW4Q 70697004 IC50 = 1700 nM T59328 C65CEI 70697160 IC50 = 2750 nM T59328 CH0B8N 70789756 IC50 > 30000 nM T59328 C5ILD4 70856339 IC50 = 91 nM T59328 CAI74T 70856585 IC50 = 10 nM T59328 C6W1NL 71244639 IC50 = 0.26 nM T59328 C5RE4T 71244643 IC50 = 0.27 nM T59328 CQ6A9L 71244644 IC50 = 0.53 nM T59328 CHT4N1 71244646 IC50 = 0.67 nM T59328 CH29GF 71258526 IC50 > 50000 nM T59328 C3BSP5 71449334 IC50 > 8000 nM T59328 C1LH2U 71449341 IC50 = 31 nM T59328 C4BXY8 71449342 IC50 = 56 nM T59328 C58BSC 71451912 IC50 = 631 nM T59328 CEBO91 71452977 IC50 = 11 nM T59328 C3MYB5 71453818 IC50 = 60 nM T59328 CJ2L8G 71455836 IC50 > 40000 nM T59328 CKT60L 71455860 Ki > 1800 nM T59328 CCGJ48 71456241 IC50 = 719 nM T59328 C7X4MD 71456750 IC50 = 10490 nM T59328 C9TZK4 71457259 IC50 = 215 nM T59328 CTWX94 71457629 IC50 > 40000 nM T59328 C3AEL4 71457630 IC50 > 40000 nM T59328 C4V6TN 71459522 IC50 > 40000 nM T59328 CEM84S 71462713 IC50 = 30 nM T59328 C7LCS8 71470563 IC50 = 12 nM T59328 CO0U6L 71473856 IC50 = 1 nM T59328 CMEH30 71473900 IC50 = 140 nM T59328 CH8NC9 71473954 IC50 = 78 nM T59328 C2PMJ7 71474167 IC50 = 4 nM T59328 CCR8J9 71496459 IC50 = 45 nM T59328 C8V4GQ 71496460 IC50 = 2 nM T59328 CQY31T 71498139 IC50 > 10000 nM T59328 C5AP8X 71508607 IC50 = 1600 nM T59328 CXQ43R 71508608 IC50 = 2200 nM T59328 CK13HD 71508609 IC50 = 1500 nM T59328 CJM0L4 71508610 IC50 = 2100 nM T59328 C2QTI4 71508643 IC50 = 8000 nM T59328 C3E4LW 71508644 IC50 = 6800 nM T59328 CQ2BV1 71508645 IC50 = 7100 nM T59328 COB85T 71508646 IC50 = 5600 nM T59328 CV6PN7 71508647 IC50 = 15300 nM T59328 CN5KQ8 71508648 IC50 = 7500 nM T59328 CDJB35 71508649 IC50 = 6100 nM T59328 CY60ZX 71508689 IC50 = 400 nM T59328 C21ZUC 71508690 IC50 = 20800 nM T59328 CSM31W 71508691 IC50 = 4600 nM T59328 C7FXT5 71508692 IC50 = 3900 nM T59328 CHZM56 71508693 IC50 = 5300 nM T59328 CK52TP 71508694 IC50 = 18600 nM T59328 C9TRM0 71508695 IC50 = 2000 nM T59328 CUHL20 71508717 IC50 = 1900 nM T59328 CY8QX5 71508718 IC50 = 4800 nM T59328 C9DIK2 71512060 IC50 = 0.2 nM T59328 C2VI1N 71512261 IC50 = 2.6 nM T59328 CF05BU 71513157 IC50 = 0.16 nM T59328 CS1ZX0 71513822 IC50 = 0.18 nM T59328 C2GP7V 71513823 IC50 = 0.89 nM T59328 CWX8Y4 71514053 IC50 = 0.3 nM T59328 CW6DN0 71514054 IC50 = 0.31 nM T59328 CXRK32 71519007 IC50 > 200 ug.mL-1 T59328 CI2Z5Y 71519008 IC50 > 200 ug.mL-1 T59328 CJ4KV6 71519009 IC50 > 200 ug.mL-1 T59328 C42MFK 71519172 IC50 > 200 ug.mL-1 T59328 C3XP1F 71519173 IC50 = 94 ug.mL-1 T59328 CC89QU 71519174 IC50 = 120 ug.mL-1 T59328 CGY2N8 71519175 IC50 > 200 ug.mL-1 T59328 C7RG1Z 71519338 IC50 = 193 ug.mL-1 T59328 COFB13 71519339 IC50 = 130 ug.mL-1 T59328 CJE5N6 71519340 IC50 = 130 ug.mL-1 T59328 CG0N8I 71519341 IC50 = 148 ug.mL-1 T59328 CM4PG6 71519493 IC50 > 200 ug.mL-1 T59328 CVUP53 71524867 IC50 = 2230 nM T59328 CQ52FW 71524868 IC50 = 8250 nM T59328 CQ7L5U 71524869 IC50 = 940 nM T59328 CVPO31 71524870 IC50 = 5680 nM T59328 CSM8Q3 71524871 IC50 = 160 nM T59328 CHZA07 71524872 IC50 = 2060 nM T59328 CW9M5E 71524873 IC50 = 210 nM T59328 C75GEB 71524914 IC50 = 3010 nM T59328 CO1H9P 71524915 IC50 = 3280 nM T59328 CNZF95 71524916 IC50 = 1070 nM T59328 CXP7G2 71524917 IC50 = 680 nM T59328 CQR8V0 71524918 IC50 = 490 nM T59328 CQ34CK 71524919 IC50 = 100 nM T59328 C12GMV 71524960 IC50 = 140 nM T59328 C7BU0K 71524961 IC50 = 300 nM T59328 C4R6CL 71524962 IC50 = 530 nM T59328 CQ7UT5 71524963 IC50 = 350 nM T59328 CRO0N8 71524964 IC50 = 1040 nM T59328 CZQ2S4 71524965 IC50 = 520 nM T59328 C8A9IN 71525006 IC50 = 660 nM T59328 CH8LC0 71525007 IC50 = 710 nM T59328 CT47DK 71525008 IC50 = 120 nM T59328 C0M4LC 71525009 IC50 = 50 nM T59328 C5OBF0 71525245 IC50 = 85900 nM T59328 CJX73B 71525246 IC50 = 110600 nM T59328 CCN90I 71525247 IC50 = 19900 nM T59328 CY6JA9 71525248 IC50 = 19300 nM T59328 CGQJ60 71525249 IC50 = 15600 nM T59328 CMKD15 71525283 IC50 = 5400 nM T59328 C3OJ6R 71525284 IC50 = 16300 nM T59328 CP5Q2U 71525285 IC50 > 200000 nM T59328 CZ8N0J 71525286 IC50 = 12800 nM T59328 CG31MI 71525287 IC50 = 26900 nM T59328 C1SFD7 71532857 IC50 > 200 ug.mL-1 T59328 C8U9MB 71532907 IC50 > 200 ug.mL-1 T59328 COQ5V1 71532908 IC50 > 200 ug.mL-1 T59328 CE9N2D 71532909 IC50 > 200 ug.mL-1 T59328 C1D3KG 71535003 Ki = 4 nM T59328 CS2X3D 71535296 Ki = 3 nM T59328 CN4AW3 71543353 IC50 = 6.1 nM T59328 CCN01X 71547862 IC50 > 10000 nM T59328 C2NLX4 71549099 IC50 = 2.7 nM T59328 CA3O6K 71552696 IC50 > 30000 nM T59328 C1NPL0 71552941 IC50 = 4290 nM T59328 CA4PS8 71552942 IC50 = 4090 nM T59328 C3UA9C 71553011 IC50 = 30000 nM T59328 CEZ15Y 71553012 IC50 = 30000 nM T59328 CVIA91 71553085 IC50 = 30000 nM T59328 C1TR3O 71553152 IC50 = 30000 nM T59328 CVNA30 71558752 IC50 > 5000 nM T59328 CEJ97M 71558906 IC50 = 600 nM T59328 C1L8GW 71558907 IC50 = 600 nM T59328 CI6QF8 71571535 IC50 = 8 nM T59328 CT4O9F 71571536 IC50 = 29 nM T59328 CRX81Q 71575642 IC50 > 10000 nM T59328 CN9BQ0 71579162 IC50 = 61 nM T59328 CN7W5S 71579325 IC50 = 126.7 nM T59328 CA9KL5 71579403 IC50 = 12.1 nM T59328 CMV9U3 71579405 IC50 = 13.6 nM T59328 C1BCX0 71579696 IC50 > 1000 nM T59328 CGK76E 71583411 IC50 > 200000 nM T59328 CB5WX0 71583412 IC50 = 42000 nM T59328 CI8K3T 71583527 IC50 = 63600 nM T59328 C6FGI0 71583528 IC50 = 38900 nM T59328 C3QGE7 71583529 IC50 > 200000 nM T59328 CS9HX7 71583530 IC50 = 114700 nM T59328 CQTZ32 71583531 IC50 = 39200 nM T59328 C0G5RS 71583532 IC50 = 58700 nM T59328 CVEY46 71583533 IC50 > 200000 nM T59328 CX6TR7 71583634 IC50 = 30800 nM T59328 CR15QP 71583635 IC50 = 130500 nM T59328 CZ31PU 71583657 IC50 = 36 nM T59328 C6RS7H 71583658 IC50 = 47 nM T59328 CWD2Z5 71585566 IC50 = 4 nM T59328 CCE7T2 71585568 IC50 = 3610 nM T59328 CO32SN 71599995 IC50 = 15 nM T59328 CQS51R 71615916 IC50 = 16 nM T59328 C4KUE9 71616518 IC50 = 56 nM T59328 CQX8L3 71616700 IC50 = 4.3 nM T59328 CE6QA1 71616701 IC50 = 3 nM T59328 C4ZDO0 71616702 IC50 = 7.4 nM T59328 C03HCR 71616703 IC50 = 0.3 nM T59328 CWTH52 71616704 IC50 = 0.5 nM T59328 CZ7XB4 71616807 IC50 = 22 nM T59328 C9YLM0 71621675 IC50 = 30 nM T59328 CH2RA9 71658877 IC50 > 5000 nM T59328 CJI05L 71658878 IC50 = 460 nM T59328 CCS41V 71658995 IC50 = 45 nM T59328 CK10SJ 71658996 IC50 > 5000 nM T59328 CI91ZX 71658997 IC50 > 5000 nM T59328 CL9T2I 71658998 IC50 > 5000 nM T59328 C1JZG9 71658999 IC50 = 1500 nM T59328 CKMO02 71659116 IC50 > 5000 nM T59328 CY5VP3 71659117 IC50 > 5000 nM T59328 CG21JR 71659118 IC50 = 2300 nM T59328 C0LHW7 71659119 IC50 = 660 nM T59328 C2IS8V 71659241 IC50 = 2500 nM T59328 C78PSE 71659242 IC50 = 3500 nM T59328 CB4LV9 71659243 IC50 = 3000 nM T59328 CGB5L8 71659244 IC50 > 5000 nM T59328 C45CVT 71659245 IC50 > 5000 nM T59328 CC6L2A 71659371 IC50 = 850 nM T59328 CQV2I4 71659372 IC50 = 900 nM T59328 CC9F0T 71659373 IC50 = 2000 nM T59328 CEBL45 71659374 IC50 = 5500 nM T59328 CHM79O 71659375 IC50 = 6000 nM T59328 CX46VT 71659505 IC50 = 5000 nM T59328 C0Y3VS 71659506 IC50 = 800 nM T59328 C3A8IH 71659507 IC50 = 1000 nM T59328 C2MS9Y 71659508 IC50 = 1500 nM T59328 C64SFQ 71659509 IC50 = 5000 nM T59328 CN6LI7 71659629 IC50 = 4500 nM T59328 C7TAL4 71659630 IC50 = 800 nM T59328 C82HXJ 71659631 IC50 = 1200 nM T59328 C2A8VJ 71659632 IC50 = 3500 nM T59328 CU27RN 71659633 IC50 = 6000 nM T59328 C2ZRK6 71659769 IC50 = 450 nM T59328 C8XM3E 71659770 IC50 = 600 nM T59328 CT79UA 71659771 IC50 = 5000 nM T59328 C6AP4D 71659772 IC50 = 6000 nM T59328 CWQ09K 71661337 IC50 = 48 nM T59328 CIK32R 71661338 IC50 = 34 nM T59328 C9PGV4 71661339 IC50 = 4327 nM T59328 CKZ6B3 71661527 IC50 > 25000 nM T59328 C1FAU8 71679855 IC50 > 100000 nM T59328 CGU2J5 71680740 IC50 = 13 nM T59328 CEWI73 71680741 IC50 = 6 nM T59328 C6K5HT 71680742 IC50 = 42 nM T59328 CFLZ59 71680901 IC50 = 20 nM T59328 CU3E6I 71680902 IC50 = 17 nM T59328 C80AGF 71680903 IC50 = 23 nM T59328 CNC9S6 71681062 IC50 = 38 nM T59328 C9TZN5 71681063 IC50 = 16 nM T59328 CT4A0M 71681064 IC50 = 101 nM T59328 CRZ1F9 71681212 IC50 = 47 nM T59328 CZ1IO5 71683105 IC50 = 14 nM T59328 CST14N 71717689 IC50 = 147 nM T59328 C1JBD5 71720447 IC50 = 4.6 nM T59328 CED2H8 71720674 IC50 = 4700 nM T59328 C30NBJ 71722055 IC50 = 2100 nM T59328 C9Z0KG 71726907 IC50 = 13 nM T59328 C4X1CP 71748056 IC50 = 874 nM T59328 C07EWM 71761646 IC50 = 17.2 nM T59328 CMO51F 71761647 IC50 = 76 nM T59328 CR08OT 71762114 IC50 = 8.4 nM T59328 CSWH95 72164480 IC50 = 4100 nM T59328 CFUD13 72164482 IC50 = 3400 nM T59328 C7P0NM 72164483 IC50 = 1500 nM T59328 C0M8QJ 72164486 IC50 = 5100 nM T59328 CD7G1S 72164602 IC50 = 4700 nM T59328 CTC7H5 72164605 IC50 = 2400 nM T59328 C5X1DO 72164726 IC50 = 3600 nM T59328 CSA2J6 72187684 IC50 = 0.677 nM T59328 CX0N2A 72189794 IC50 = 0.63 nM T59328 CZ3XL6 72190112 IC50 = 0.41 nM T59328 CSK78J 72190113 IC50 = 19 nM T59328 CF4TJ9 72191350 IC50 = 190 nM T59328 CP2OR8 72191351 IC50 = 52 nM T59328 CM1B2Y 72191352 IC50 = 158 nM T59328 C5L0BJ 72191353 IC50 = 26 nM T59328 C4J3KE 72191667 IC50 = 94 nM T59328 C4DQ3P 72191668 IC50 = 36 nM T59328 C1YC7S 72191669 IC50 = 48 nM T59328 CNMJ61 72191670 IC50 = 24 nM T59328 C2MQ6X 72191671 IC50 = 25 nM T59328 CEB67M 72191672 IC50 = 34 nM T59328 C7V8MX 72195043 IC50 = 6 nM T59328 C1R7VY 72195184 IC50 = 8.1 nM T59328 CQR2N5 72201345 IC50 = 1.2 nM T59328 CC2X5T 72201349 IC50 = 0.5 nM T59328 CF75TB 72201501 IC50 = 4 nM T59328 CFA2J9 72201502 IC50 = 6.7 nM T59328 CIU90H 72202607 IC50 = 16 nM T59328 C4N9OI 72202732 IC50 = 1.07 nM T59328 CKAF40 72202733 IC50 = 33885 nM T59328 C7FJB9 72202734 IC50 = 13.8 nM T59328 CSW20D 72202735 IC50 = 4.53 nM T59328 CYB05D 72202865 IC50 = 3.97 nM T59328 C2MY1Q 72202866 IC50 = 6754 nM T59328 CV23JN 72202867 IC50 = 4.96 nM T59328 CW8HV3 72202868 IC50 = 4.72 nM T59328 C6FZA2 72202870 IC50 = 17.6 nM T59328 COK12B 72202930 IC50 = 0.5 nM T59328 CI3B4N 72202931 IC50 = 0.2 nM T59328 C8WC6P 72202999 IC50 = 4.94 nM T59328 C1TIX3 72203001 IC50 = 60.4 nM T59328 CW18BO 72203003 IC50 = 6.95 nM T59328 CI63WE 72203004 IC50 = 691 nM T59328 CYT82Q 72203134 IC50 = 39.7 nM T59328 C0K6SQ 72203136 IC50 = 26283 nM T59328 C7MV3O 72203732 IC50 = 250 nM T59328 CYB30W 72203733 IC50 = 410 nM T59328 C90ZBE 72203734 IC50 = 19 nM T59328 C5EWB0 72203735 IC50 = 68 nM T59328 C6KB7T 72203914 IC50 = 45 nM T59328 C9Q6LM 72206524 IC50 = 780 nM T59328 CKH1F8 72206525 IC50 = 960 nM T59328 CUT5W6 72206526 IC50 = 140 nM T59328 CE1VK7 72543781 IC50 = 13200 nM T59328 CLM4G2 72543782 IC50 = 9800 nM T59328 CF9LG1 72543783 IC50 = 31400 nM T59328 C3AT2E 72543784 IC50 = 3100 nM T59328 C32RMJ 72544014 IC50 = 7400 nM T59328 C7J4XV 72544015 IC50 = 6500 nM T59328 CPL35N 72544251 IC50 = 7600 nM T59328 CNT79J 72545791 IC50 = 10020 nM T59328 CN89UW 72545792 IC50 = 6130 nM T59328 CGY75C 72545793 IC50 = 12450 nM T59328 C8U6KH 72546029 IC50 = 2580 nM T59328 CW4VL8 72546030 IC50 = 1890 nM T59328 COR35N 72546031 IC50 = 210 nM T59328 CC9VQ1 72546032 IC50 = 430 nM T59328 C5QZS6 72546033 IC50 = 8190 nM T59328 CAM91I 72547360 IC50 = 8100 nM T59328 CEZQ57 72697432 IC50 = 1230 nM T59328 CL7A4Z 72697433 IC50 = 1180 nM T59328 CUD9M1 72697435 IC50 = 3510 nM T59328 C4AWS3 72697576 IC50 = 5490 nM T59328 C5M3GE 72697580 IC50 = 2120 nM T59328 COX45Z 72697720 IC50 = 3060 nM T59328 C10VYB 72697722 IC50 = 1380 nM T59328 CJ7E1C 72699656 IC50 = 4 nM T59328 CF4D5O 72699657 IC50 = 10 nM T59328 C52NAB 72699658 IC50 > 50000 nM T59328 C64UEN 72699659 IC50 > 32770 nM T59328 CKPL31 72700004 IC50 = 6810 nM T59328 C90VOI 72700006 IC50 = 50 nM T59328 CA4M7U 72700007 IC50 > 50000 nM T59328 CWZG30 72700008 IC50 > 50000 nM T59328 CG7AI6 72700079 IC50 > 50000 nM T59328 CI8ZY3 72700080 IC50 > 50000 nM T59328 CWRL78 72700165 IC50 = 4 nM T59328 CWBC84 72703789 IC50 = 421 nM T59328 CM75FY 72703989 IC50 = 68 nM T59328 CPQ34Z 72703991 IC50 = 72 nM T59328 CYG95S 72707651 IC50 > 5000 nM T59328 CNP0V5 72707724 IC50 > 5000 nM T59328 CU4A5Q 72707728 IC50 > 5000 nM T59328 CZAM98 72707790 IC50 > 5000 nM T59328 CP13FK 72707853 IC50 > 5000 nM T59328 C9OQ2I 72710839 IC50 > 10000 nM T59328 C26NTQ 72712708 IC50 = 708.5 nM T59328 CBN20W 72712709 IC50 = 143.6 nM T59328 C1XO0R 72712710 IC50 > 1000 nM T59328 CQ96FB 72712711 IC50 = 525 nM T59328 CEF73D 72712712 IC50 = 864 nM T59328 C4BX2Y 72712713 IC50 = 58.7 nM T59328 C01QBS 72712714 IC50 = 42.9 nM T59328 CAZ9P0 72712883 IC50 = 40.3 nM T59328 CA26ZY 72712884 IC50 = 204.1 nM T59328 CVH9B7 72712885 IC50 = 107.1 nM T59328 C9R5TW 72712886 IC50 = 8.8 nM T59328 CWI13Y 72712887 IC50 = 15.2 nM T59328 C9F8WM 72712888 IC50 = 235.4 nM T59328 CO7YX5 72712889 IC50 = 29.1 nM T59328 C2GRZ1 72712890 IC50 = 97.9 nM T59328 CX9L1B 72712891 IC50 = 16.2 nM T59328 C8R5SM 72712892 IC50 = 41.3 nM T59328 CRI42Q 72712893 IC50 = 7.2 nM T59328 CLX3M1 72712894 IC50 = 17.1 nM T59328 CSNU50 72712895 IC50 = 55.5 nM T59328 C54LQO 72712896 IC50 = 35.6 nM T59328 CY56SR 72712897 IC50 = 9.2 nM T59328 CUS2R1 72712978 IC50 = 21280 nM T59328 C87MUD 72712979 IC50 = 3836 nM T59328 C5ZU4Y 72713172 IC50 = 4802 nM T59328 CUDS15 72713174 IC50 = 31.3 nM T59328 CH93FM 72713175 IC50 = 373.5 nM T59328 CH3K0R 72713176 IC50 = 5585 nM T59328 C9LA5P 72713177 IC50 = 5.12 nM T59328 CK3N8G 72713385 IC50 = 272 nM T59328 CXU6R4 72713386 IC50 = 16338 nM T59328 CGN60W 72713387 IC50 = 5.29 nM T59328 CPA37Q 72734868 IC50 = 464 nM T59328 CJE91U 72734869 IC50 = 699 nM T59328 C2ZP3W 72734870 IC50 = 859 nM T59328 CWQ1G5 72734871 IC50 = 884 nM T59328 C0AVR4 72734872 IC50 = 1715 nM T59328 CSDQ79 72735047 IC50 = 265 nM T59328 CW3HI2 72735048 IC50 = 304 nM T59328 CG82VX 72735049 IC50 = 331 nM T59328 CKU16J 72735050 IC50 = 232 nM T59328 CFM8W4 72735051 IC50 = 404 nM T59328 CI2YH8 72737033 IC50 = 27 nM T59328 CE7T5Y 72737034 IC50 = 479 nM T59328 CIDN27 72737035 IC50 = 41 nM T59328 CTC3I9 72737206 IC50 = 635 nM T59328 C6QFZ8 72737207 IC50 = 365 nM T59328 C60TUV 72737208 IC50 = 68 nM T59328 CZ7U9H 72737209 IC50 = 165 nM T59328 CNX58O 72737210 IC50 = 82 nM T59328 CZ4IY1 72737401 IC50 = 197 nM T59328 CC38YI 72737402 IC50 = 544 nM T59328 C4SRQ7 72737403 IC50 = 24 nM T59328 CJ3WA6 72737404 IC50 = 32 nM T59328 CL7WI5 72737405 IC50 = 281 nM T59328 C8ADG7 72737575 IC50 = 505 nM T59328 CU9PS0 72737576 IC50 = 464 nM T59328 C8IV1S 72737577 IC50 = 543 nM T59328 C2S1ZE 72737578 IC50 = 967 nM T59328 C20NFB 72737579 IC50 = 1581 nM T59328 CQF4K5 72950786 IC50 = 0.79 nM T59328 CP58UB 73053605 IC50 = 3 nM T59328 C89HEJ 73291830 IC50 = 250 nM T59328 C5LGB4 73291831 IC50 = 220 nM T59328 CWC12F 73291832 IC50 = 290 nM T59328 C4B1CL 73291833 IC50 = 15200 nM T59328 CG8RI0 73292361 IC50 = 19 nM T59328 CC16IJ 73292362 IC50 = 19000 nM T59328 C7LPO0 73292363 IC50 = 5.6 nM T59328 CBQ72N 73292545 IC50 = 63 nM T59328 C9M7EL 73294313 IC50 = 770 nM T59328 CED6P2 73294314 IC50 = 81 nM T59328 CTPF92 73294315 IC50 = 22 nM T59328 C87AQU 73294502 IC50 = 12900 nM T59328 CDM86C 73294503 IC50 = 2100 nM T59328 C0D5EA 73294504 IC50 = 2800 nM T59328 C2UB8T 73294505 IC50 = 33 nM T59328 CAU94B 73294506 IC50 = 1550 nM T59328 CQV1P0 73294507 IC50 = 91 nM T59328 C3MF2U 73335400 IC50 = 9 nM T59328 C3QEG6 73335403 IC50 = 72 nM T59328 CE25BK 73335501 IC50 = 27 nM T59328 CZ90QC 73335502 IC50 = 32 nM T59328 CZP84O 73335598 IC50 > 10000 nM T59328 CJ3BK2 73335600 IC50 = 34 nM T59328 C06IFC 73335691 IC50 = 390 nM T59328 CC4DW1 73335692 IC50 = 33 nM T59328 C9JS7Z 73335693 IC50 = 880 nM T59328 C43EUZ 73335785 IC50 = 27 nM T59328 C0HSC8 73346520 Ki = 6090 nM T59328 C8SD9P 73346521 Ki = 55290 nM T59328 CGZ6Y8 73346522 Ki = 6640 nM T59328 C18WCY 73346557 IC50 = 1.29 nM T59328 C41QZC 73347162 Ki = 4000 nM T59328 C43IPQ 73348006 Ki = 15650 nM T59328 C8SIL6 73349435 IC50 = 90.05 nM T59328 CV21FR 73349643 IC50 = 100 nM T59328 C9EXR4 73351100 IC50 = 21.1 nM T59328 CS9C0W 73351108 Ki = 27400 nM T59328 CXC0O2 73352566 IC50 = 25.1 nM T59328 CZJ2S7 73352567 IC50 = 18.7 nM T59328 CCI47S 73352568 IC50 = 10.8 nM T59328 C27JUH 73352576 Ki = 8580 nM T59328 CVP03Z 73352577 Ki = 41580 nM T59328 CX75YR 73352604 IC50 = 630.96 nM T59328 C9TMA1 73352657 IC50 = 100 nM T59328 CDAB86 73354065 Ki = 2970 nM T59328 CK3Z8U 73354066 Ki = 4680 nM T59328 C92DXZ 73354067 Ki = 22940 nM T59328 C83XBD 73354112 IC50 = 7 nM T59328 CCI18Y 73355591 Ki = 5820 nM T59328 CRX8A0 73355592 Ki = 16770 nM T59328 C8XHK6 73356867 IC50 = 2300 nM T59328 CYQ8K1 73357210 IC50 = 70 nM T59328 CVNW01 73386831 IC50 > 1000 nM T59328 CQ5E3H 73707531 IC50 = 16.8 nM T59328 CX1LR9 73774633 IC50 = 26 nM T59328 CS9BQ1 74222426 IC50 = 3890 nM T59328 CO0V6K 74222427 IC50 = 16800 nM T59328 CBE71O 74222509 IC50 > 20000 nM T59328 CM02PA 74222510 IC50 = 1710 nM T59328 CWLT81 74222511 IC50 > 20000 nM T59328 C4XSG8 74222512 IC50 = 274 nM T59328 CBT4M6 74222513 IC50 = 2180 nM T59328 C53AFH 74222599 IC50 = 2910 nM T59328 CNR7C1 74223711 IC50 = 126.3 nM T59328 CJ0N5V 74223816 IC50 = 1.06 nM T59328 CF9A7B 74766095 Ki = 2 nM T59328 CM1VR8 74766099 Ki = 0.14 nM T59328 C4WHJ6 74937126 IC50 = 1 nM T59328 C97KTL 76007179 IC50 = 34.16 nM T59328 C7K2QN 76280903 Ki = 22 nM T59328 CP1W6F 76281713 Ki = 151 nM T59328 CN1RJ8 76282701 Ki = 18 nM T59328 C1XZY3 76282702 Ki = 14 nM T59328 CFP9O7 76309779 IC50 = 7300 nM T59328 CW5OG2 76310006 IC50 = 61500 nM T59328 C8DX4U 76311274 IC50 = 275 nM T59328 C0HX2E 76311275 IC50 = 53300 nM T59328 C07IBW 76312208 IC50 = 250034.54 nM T59328 CH24LB 76313481 IC50 = 130 nM T59328 C7MLX4 76313718 IC50 = 18300 nM T59328 CRV24X 76313719 IC50 > 100000 nM T59328 CW5A6P 76314206 IC50 > 10000 nM T59328 CDG1O5 76316997 IC50 = 200 nM T59328 C0M2LJ 76316998 IC50 = 1100 nM T59328 CZK2V6 76317238 IC50 > 100000 nM T59328 CKG8C3 76317239 IC50 = 34600 nM T59328 C27JRQ 76317764 IC50 = 4 nM T59328 C8AJ3M 76317765 IC50 = 3 nM T59328 C4PT8M 76318480 IC50 > 5000 nM T59328 CF06PR 76318481 IC50 = 2200 nM T59328 CK5UL0 76318482 IC50 = 2000 nM T59328 CE95GB 76318483 IC50 = 43700 nM T59328 CX7RD0 76320712 IC50 = 1200 nM T59328 CJE4B1 76321478 IC50 = 16 nM T59328 C13XBM 76321479 IC50 > 10000 nM T59328 CG29RA 76321480 IC50 > 10000 nM T59328 CLO8N7 76321481 IC50 > 10000 nM T59328 CG67DB 76321482 IC50 = 12 nM T59328 C6SCV7 76322145 IC50 = 3200 nM T59328 CL0T7B 76322219 IC50 = 2145 nM T59328 CPD3W5 76324607 IC50 = 1630 nM T59328 CZ6AK2 76325089 IC50 > 10000 nM T59328 CBP83A 76325766 IC50 = 2.1 nM T59328 C4K7IO 76325767 IC50 = 2300 nM T59328 C4RD8T 76325768 IC50 = 1.5 nM T59328 CH6V0B 76327248 IC50 = 12880 nM T59328 CHDR08 76327920 IC50 = 9 nM T59328 CPZN18 76328168 IC50 > 100000 nM T59328 CDP53X 76328653 IC50 > 10000 nM T59328 CE1L8A 76329348 IC50 = 931 nM T59328 CV4ZP1 76331568 IC50 = 33 nM T59328 CA45HZ 76331569 IC50 = 3 nM T59328 C0BJ8F 76332331 IC50 = 5 nM T59328 C83DTC 76332332 IC50 > 10000 nM T59328 CJ2T9E 76332983 IC50 = 270 nM T59328 CC25SV 76332992 IC50 = 9800 nM T59328 CS47NK 76332993 IC50 = 2800 nM T59328 C7K1PL 76332994 IC50 = 3950 nM T59328 COTE80 76332995 IC50 = 2500 nM T59328 C9GRT4 76332996 IC50 = 76500 nM T59328 CAP7F0 76335418 IC50 = 67200 nM T59328 C51LIY 76335419 IC50 > 100000 nM T59328 C4J5BS 76335961 IC50 = 5 nM T59328 C28UES 76335962 IC50 > 10000 nM T59328 CG56FE 76335963 IC50 = 82 nM T59328 CP3YE6 76336599 IC50 = 3710 nM T59328 C4V0GX 76336600 IC50 = 4400 nM T59328 CZR21Q 76336601 IC50 = 8730 nM T59328 C4QPA1 76336602 IC50 = 130 nM T59328 C2N9EB 76336603 IC50 = 2200 nM T59328 C4HOM3 76900440 IC50 = 1935 nM T59328 CT92YM 77461033 IC50 = 6 nM T59328 CH8W7D 77461036 IC50 > 1000 nM T59328 CWG4T2 78209992 IC50 < 0.5 nM T59328 CS8V1X 78318941 IC50 = 2.9 nM T59328 CA5SQ8 78319175 IC50 = 1 nM T59328 CH8XY3 78322920 IC50 > 10000 nM T59328 C2YSJ7 78323235 IC50 > 10000 nM T59328 CTJ02F 78323236 IC50 > 10000 nM T59328 C5P4JF 78323237 IC50 > 10000 nM T59328 CVZ26O 78323238 IC50 > 10000 nM T59328 CP90IE 78323239 IC50 = 890 nM T59328 CAZ2J6 78323563 IC50 = 1010 nM T59328 CXC01P 78323564 IC50 = 360 nM T59328 CGP5M8 78323565 IC50 > 10000 nM T59328 CNA52Z 78324176 IC50 = 9 nM T59328 C90PJT 78324177 IC50 = 3 nM T59328 CEDG87 78324478 IC50 = 5 nM T59328 C2JKT5 78324480 IC50 = 27 nM T59328 CQA2Y0 78324481 IC50 = 3 nM T59328 CT81NA 78324482 IC50 = 550 nM T59328 CV0P3A 78357783 IC50 = 200 nM T59328 C7CGZ1 85206710 IC50 = 800 nM T59328 CK61HY 85469442 IC50 > 10000 nM T59328 CL19KE 85471023 IC50 = 5.3 nM T59328 CYAS09 85471025 IC50 = 2.1 nM T59328 C93JAB 85471026 IC50 = 520.2 nM T59328 C97GER 85471045 IC50 = 356.6 nM T59328 C7YK6I 85471046 IC50 = 109.4 nM T59328 CD51LP 85471121 IC50 = 1.56 nM T59328 CRT9W7 85471122 IC50 = 1.3 nM T59328 CNXC02 85471147 IC50 = 4.5 nM T59328 CR1O7P 85471149 IC50 = 3.5 nM T59328 C2WLZ6 85827467 Ki = 700 nM T59328 CV4TL7 86276219 IC50 = 270 nM T59328 CH2X3O 86276220 IC50 = 21020 nM T59328 C8R4JZ 86276226 IC50 = 4100 nM T59328 CRA39W 86276227 IC50 = 180 nM T59328 C7QXC2 86276228 IC50 = 120 nM T59328 C7GE4I 86276229 IC50 = 420 nM T59328 CBQ9L7 86276271 IC50 < 0.25 nM T59328 CQ9H4U 86277844 IC50 = 7500 nM T59328 CV8UZ1 86278565 Ki = 17 nM T59328 CSH3G2 86287525 IC50 > 10000 nM T59328 C0QK9F 86288869 IC50 = 94 nM T59328 CWYE62 86294833 IC50 = 1320 nM T59328 CCJ43A 86302281 IC50 = 16 nM T59328 CH5AD6 86302282 IC50 = 9 nM T59328 CJL1W6 86302308 IC50 = 4 nM T59328 C7U3VF 86302309 IC50 = 3 nM T59328 CA72QE 86302441 IC50 = 510 nM T59328 CQ9J7S 86302442 IC50 = 10120 nM T59328 CB5NJ4 86302541 IC50 > 10000 nM T59328 CPG3A5 86302574 IC50 > 30000 nM T59328 C7MA0Y 86302767 IC50 = 444.7 nM T59328 C2L4GR 86303858 IC50 = 4 nM T59328 C08WGI 86566799 IC50 > 10000 nM T59328 C9NTP1 86677234 IC50 = 2000 nM T59328 CEKQ13 86677242 IC50 = 19000 nM T59328 C5YX8T 86677253 IC50 = 1000 nM T59328 CCX1U5 86677265 IC50 = 2000 nM T59328 CZQ1F7 86677270 IC50 = 311 nM T59328 CB5Z8H 86677276 IC50 < 1 nM T59328 C1KLC3 86679616 Ki = 3 nM T59328 CR08QT 89266687 IC50 = 550 nM T59328 CNZ86G 89456691 IC50 = 7.6 nM T59328 CP0MJ8 89456904 Ki = 35 nM T59328 CK78NF 89456980 Ki = 3 nM T59328 CY12PC 89457089 Ki = 8 nM T59328 CS42DR 89457109 Ki = 8 nM T59328 C32JOH 89457151 Ki = 4 nM T59328 C1HTP4 89457165 Ki = 4 nM T59328 CNSK27 89457251 Ki = 3 nM T59328 CR5QA1 89457296 IC50 = 1.6 nM T59328 CM8T1V 89556219 IC50 = 36 nM T59328 C1HW4B 89735655 IC50 > 100000 nM T59328 CR3XL7 90119070 IC50 > 20000 nM T59328 CLK3O0 90119255 IC50 = 570 nM T59328 CO2FV0 90119264 IC50 = 15 nM T59328 C3RL4C 90136268 IC50 > 20000 nM T59328 C4ME0V 90136282 IC50 = 15400 nM T59328 CY0T6O 90136348 IC50 = 149 nM T59328 CN2RJ1 90178371 Ki = 20 nM T59328 C5XEP6 90183257 Ki = 76 nM T59328 C70HZA 90183266 Ki = 201 nM T59328 C3G4AS 90183295 Ki = 149 nM T59328 CM6GB2 90183305 Ki = 19 nM T59328 C4DEJ1 90183313 Ki = 71 nM T59328 CHR3J1 90183333 Ki = 48 nM T59328 C70EWF 90183350 Ki = 87 nM T59328 CV64KY 90183363 Ki = 40 nM T59328 C1GZ4H 90183367 Ki = 19 nM T59328 CY3P2G 90183439 Ki = 124 nM T59328 CKQ87S 90183468 Ki = 27 nM T59328 C5HZ0I 90183471 Ki = 658 nM T59328 CIR8P9 90183483 Ki = 28 nM T59328 CD08SZ 90183490 Ki = 196 nM T59328 CL12RI 90183503 Ki = 323 nM T59328 C8NLP0 90183548 Ki = 329 nM T59328 C97YQB 90183560 Ki = 2.7 nM T59328 C7TQI0 90183635 Ki = 492 nM T59328 C7TKR1 90183640 Ki = 77 nM T59328 C03ZHC 90183641 Ki = 24 nM T59328 C9A4WX 90183658 Ki = 2.5 nM T59328 CR7CN0 90183696 Ki = 38 nM T59328 CON0U4 90183732 Ki = 50 nM T59328 CL4JO2 90183809 Ki = 33 nM T59328 C7DT2U 90183870 Ki > 0.53 nM T59328 C8BJ6V 90183913 Ki = 4.3 nM T59328 CX4L6E 90183992 Ki = 13 nM T59328 CWT70U 90185859 IC50 = 94 nM T59328 CZF18X 90185862 IC50 = 11 nM T59328 CAF0J8 90185892 IC50 = 1.3 nM T59328 C2QD8N 90185907 IC50 = 10 nM T59328 CIY1J5 90185909 IC50 = 19 nM T59328 CIT45C 90185926 IC50 = 39 nM T59328 CA6KX8 90185944 IC50 = 95 nM T59328 CK2NU8 90185982 IC50 = 78 nM T59328 C75IJT 90185983 IC50 = 23.5 nM T59328 CLT57U 90185984 IC50 = 20 nM T59328 CS6VQ3 90186050 IC50 = 17.8 nM T59328 CB9CG5 90282624 IC50 = 1 nM T59328 CPH85G 90322858 IC50 = 4 nM T59328 C1UQ3H 90375291 IC50 = 1.2 nM T59328 CF7XO6 90375389 IC50 = 63.8 nM T59328 C5S3YB 90645165 IC50 > 10000 nM T59328 CY0UC4 90645194 IC50 > 10000 nM T59328 C3GU7P 90645237 IC50 > 10000 nM T59328 CFI93O 90645239 IC50 > 10000 nM T59328 C76KSB 90645241 IC50 > 10000 nM T59328 CNWP80 90645243 IC50 > 10000 nM T59328 C1POJ2 90645244 IC50 > 10000 nM T59328 C8BEX4 90645245 IC50 > 10000 nM T59328 C6Q4DH 90645475 IC50 = 73.3 nM T59328 C89HTB 90645476 IC50 = 340.1 nM T59328 CL32MR 90645477 IC50 = 113.2 nM T59328 C9ASG1 90645478 IC50 = 70.7 nM T59328 COY53U 90645479 IC50 = 30 nM T59328 C48OSQ 90645480 IC50 = 84.4 nM T59328 CL8GW5 90645481 IC50 = 122.1 nM T59328 CL7SC6 90645482 IC50 = 90.2 nM T59328 C5U6RM 90645483 IC50 = 30.2 nM T59328 CI3OD6 90645484 IC50 = 42.2 nM T59328 CCS47U 90645485 IC50 = 145.2 nM T59328 CXEB69 90645486 IC50 = 102.3 nM T59328 CX29IY 90655145 IC50 = 4 nM T59328 CI56KC 90655146 IC50 > 10000 nM T59328 C5LI2K 90655147 IC50 > 10000 nM T59328 C7J3GQ 90655148 IC50 > 10000 nM T59328 CG09KP 90655149 IC50 = 4997 nM T59328 CJ6EV4 90655150 IC50 > 10000 nM T59328 CE9V5Z 90655151 IC50 = 799 nM T59328 CZ5U8S 90655152 IC50 = 4286 nM T59328 CCFD23 90655153 IC50 = 1699 nM T59328 C3ZFB7 90655154 IC50 = 542 nM T59328 C1NIF5 90655155 IC50 = 3399 nM T59328 C0OIN4 90655156 IC50 = 770 nM T59328 C8O2FA 90655157 IC50 = 6414 nM T59328 CNKM05 90655158 IC50 = 1792 nM T59328 CT7V5Z 90655159 IC50 = 40 nM T59328 CC4M2L 90655160 IC50 = 5 nM T59328 CT4U7R 90655161 IC50 = 1196 nM T59328 CWTH01 90655162 IC50 = 68 nM T59328 C8H7MU 90655163 IC50 = 10 nM T59328 CX2KS1 90655164 IC50 = 20 nM T59328 C5YLC2 90655165 IC50 = 8 nM T59328 CKW2E0 90655166 IC50 = 24 nM T59328 CR9G6B 90655167 IC50 = 8 nM T59328 CW7H2X 90655168 IC50 = 2 nM T59328 CZ2G8V 90655169 IC50 = 139 nM T59328 C3VR8U 90655170 IC50 = 93 nM T59328 C8T9EB 90655171 IC50 = 38 nM T59328 CIW07X 90655172 IC50 = 28 nM T59328 C9D3JH 90655173 IC50 = 4 nM T59328 C8AS4G 90655174 IC50 = 18 nM T59328 CJS7X5 90655175 IC50 = 3 nM T59328 CJ5BC8 90655176 IC50 = 4 nM T59328 CC6BI4 90655177 IC50 = 34 nM T59328 C0ZEA7 90655178 IC50 = 7 nM T59328 CJ6ZX7 90655179 IC50 = 7 nM T59328 CH8QP2 90655180 IC50 = 2159 nM T59328 CI0TR8 90655181 IC50 = 2 nM T59328 CY9FE6 90655275 IC50 = 550 nM T59328 C1CFP6 90655276 IC50 = 575 nM T59328 CI8XW3 90655277 IC50 > 10000 nM T59328 CT28VM 90655278 IC50 > 10000 nM T59328 C8N5TF 90655279 IC50 = 3900 nM T59328 CPN1I6 90655280 IC50 = 1920 nM T59328 CW1LJ4 90655281 IC50 = 43 nM T59328 CAC3D4 90655282 IC50 = 1330 nM T59328 CKO3Z1 90655283 IC50 = 120 nM T59328 C7S8KR 90655284 IC50 = 130 nM T59328 CY0T9O 90655285 IC50 = 43 nM T59328 CG9HX4 90655286 IC50 = 44 nM T59328 C7DT3G 90655287 IC50 = 33 nM T59328 C8RA1Y 90655288 IC50 = 47 nM T59328 C1B7TW 90655289 IC50 = 6 nM T59328 CVO26Z 90655290 IC50 = 5540 nM T59328 CO5M8T 90655291 IC50 = 30 nM T59328 CXNB56 90655292 IC50 > 10000 nM T59328 CW08SL 90655293 IC50 = 680 nM T59328 CC2P7K 90655294 IC50 = 99 nM T59328 CBX47C 90655295 IC50 = 160 nM T59328 CEDA08 90655430 IC50 = 88 nM T59328 C8ZUA3 90655431 IC50 = 877 nM T59328 C82SHX 90655432 IC50 = 184 nM T59328 CEY4A8 90655433 IC50 = 2177 nM T59328 CX5E6G 90655434 IC50 > 10000 nM T59328 COQ34Y 90655435 IC50 = 4706 nM T59328 CPXQ71 90655436 IC50 = 537 nM T59328 C56FLY 90655437 IC50 = 2388 nM T59328 CIQ9S0 90655438 IC50 = 201 nM T59328 C0LFA1 90655439 IC50 = 18020 nM T59328 C3IZ1H 90655440 IC50 = 4150 nM T59328 CT52QD 90655441 IC50 = 32130 nM T59328 C2JX1T 90655442 IC50 = 14700 nM T59328 C2Q1FV 90655443 IC50 = 24050 nM T59328 CR8CQ1 90655444 IC50 = 2090 nM T59328 C4HB6Y 90655445 IC50 = 910 nM T59328 CC76UY 90655446 IC50 = 6150 nM T59328 CC8BR4 90655447 IC50 = 11180 nM T59328 C2BD4K 90655448 IC50 = 1030 nM T59328 C8BL6E 90655679 IC50 = 1580 nM T59328 C2Z7EO 90655680 IC50 = 8660 nM T59328 CAB7E0 90655681 IC50 = 10350 nM T59328 CO8PA3 90655682 IC50 = 7670 nM T59328 C0S1HF 90655767 IC50 > 16000 nM T59328 CW5ZR6 90655768 IC50 = 7670 nM T59328 C51MOA 90655769 IC50 = 3860 nM T59328 CZ6U5W 90655770 IC50 = 1370 nM T59328 C7P6FQ 90655771 IC50 = 84 nM T59328 CXA18Y 90655772 IC50 = 168 nM T59328 C15GJU 90655773 IC50 = 572 nM T59328 C25CWH 90655774 IC50 = 4354 nM T59328 CFRI21 90655775 IC50 = 1201 nM T59328 CAIL45 90655776 IC50 = 1052 nM T59328 CVYA67 90655777 IC50 = 1907 nM T59328 CA84HG 90656352 IC50 = 3960 nM T59328 CW2Z7O 90656353 IC50 = 5530 nM T59328 C0CZ6J 90656354 IC50 = 5260 nM T59328 CRO40H 90656355 IC50 = 650 nM T59328 CQF9S2 90656356 IC50 = 6310 nM T59328 CU12BF 90656357 IC50 = 2800 nM T59328 CO5F7S 90656358 IC50 = 3250 nM T59328 C3PT4O 90656359 IC50 = 120 nM T59328 CP34KC 90664681 IC50 = 1910 nM T59328 CK3IS4 90664930 IC50 = 2280 nM T59328 CRL86F 90665697 IC50 = 650 nM T59328 CR34GP 90666149 IC50 = 9.14 nM T59328 C3RK6C 90666150 IC50 > 1000 nM T59328 CXB1P6 90666151 IC50 = 2.45 nM T59328 CE3VO1 90666152 IC50 = 22.12 nM T59328 C1QYH8 90666153 IC50 = 24.83 nM T59328 C3Q2OD 90666154 IC50 = 10.18 nM T59328 C6CD0G 90666155 IC50 = 77.19 nM T59328 CR1A3V 90666156 IC50 = 6.99 nM T59328 CE6B1Q 90666157 IC50 = 4.68 nM T59328 CP9O1K 90666158 IC50 = 33.95 nM T59328 CSQ89J 90666159 IC50 = 37.37 nM T59328 CF4VN5 90666317 IC50 = 5.78 nM T59328 CNSL72 90666318 IC50 = 6.26 nM T59328 C9V6FU 90666397 IC50 = 520 nM T59328 C5Q8VO 90666398 IC50 = 590 nM T59328 CIB1E8 90666399 IC50 = 570 nM T59328 C08ANK 90666400 IC50 = 800 nM T59328 CL0KH2 90666401 IC50 = 460 nM T59328 C9XI3E 90666402 IC50 = 510 nM T59328 CLF29C 90666403 IC50 > 1000 nM T59328 CU9XB7 90666404 IC50 > 1000 nM T59328 CCL19D 90666405 IC50 > 1000 nM T59328 CYVM38 90666406 IC50 > 1000 nM T59328 CMY4T0 90666407 IC50 > 1000 nM T59328 CNE54X 90666408 IC50 > 1000 nM T59328 CBAM42 90667697 IC50 > 10000 nM T59328 C3TCZ8 90667699 IC50 > 10000 nM T59328 C1M7UL 90667701 IC50 > 10000 nM T59328 C7J0CF 90667703 IC50 > 10000 nM T59328 CU5I7B 90667705 IC50 > 10000 nM T59328 CH16WR 90667707 IC50 > 10000 nM T59328 C8SX2E 90667875 IC50 = 8000 nM T59328 CS73QB 90667877 IC50 = 3900 nM T59328 CSM40E 90667879 IC50 > 10000 nM T59328 CAZD95 90667881 IC50 = 8500 nM T59328 CGU4Q0 90667883 IC50 = 5500 nM T59328 CN1L2V 90667885 IC50 > 10000 nM T59328 C96DTL 90682879 IC50 = 82.3 nM T59328 CF6Q9X 91669170 IC50 = 90 nM T59328 COWV98 91844461 IC50 = 700 nM T59328 C51PJL 91864590 IC50 = 4 nM T59328 C0Y8ZK 91933875 IC50 > 1000 nM T59328 CQTF61 91970514 IC50 = 1600 nM T59328 CE4Q5N 91970515 IC50 = 3900 nM T59328 CC23OD 91970516 IC50 = 900 nM T59328 CB8AR9 91970527 IC50 > 10000 nM T59328 C70ZPT 91971390 Ki = 64 nM T59328 CGQ95X 91971392 Ki = 52 nM T59328 CAU45T 91971978 IC50 > 30000 nM T59328 C64SIO 92042864 IC50 = 409 nM T59328 CWF97Y 92045039 IC50 = 3 nM T59328 C8F7XO 92131166 IC50 = 529.4 nM T59328 CVZ65G 92132732 Ki = 1.5 nM T59328 CMZ92J 92132733 Ki = 1.1 nM T59328 C4CE3S 94146587 IC50 = 34280 nM T59328 CC1Q3Y 95171151 IC50 > 10000 nM T59328 CR02CX 95171152 IC50 = 38 nM T59328 CO4GL7 101879115 IC50 = 0.47 nM T59328 C05NTY 101884761 IC50 = 938000 nM T59328 CWM71R 101884762 IC50 = 600 nM T59328 CRI0S4 101891768 Ki = 12 nM T59328 CK72FW 102129497 IC50 > 10000 nM T59328 CQ7B8D 102515536 Ki = 37 nM T59328 C9SF3U 102515537 Ki = 4 nM T59328 C9G5TC 102515538 Ki = 19 nM T59328 C78NRU 112865697 IC50 = 208 nM T59328 CI6H8C 112865788 IC50 = 974 nM T59328 COU61I 112865858 IC50 = 901 nM T59328 CIR97O 112866175 IC50 = 7.7 nM T59328 C2BAR8 112866205 IC50 = 1188 nM T59328 CU4O5Z 112901888 IC50 = 11000 nM T59328 CM7C3W 117668218 IC50 = 5.9 nM T59328 CTK65N 117668270 IC50 = 208 nM T59328 C63LHQ 117668291 IC50 = 2.2 nM T59328 C0V3ZB 117676956 IC50 < 0.25 nM T59328 CO4Z3X 117676961 IC50 < 0.25 nM T59328 C7RUS2 117676973 IC50 < 0.25 nM T59328 C3NI4J 117676976 IC50 < 0.25 nM T59328 C5LWU4 117677006 IC50 < 0.25 nM T59328 CO01EN 117780037 IC50 = 3 nM T59328 C30HQS 117780120 IC50 = 1860 nM T59328 C2DEK4 117780234 IC50 = 1.5 nM T59328 C5FD2M 117803130 IC50 = 5 nM T59328 CLQ3I0 117803131 IC50 = 6 nM T59328 C21MWK 117803134 IC50 = 2 nM T59328 CX6LJ9 117803651 IC50 = 6 nM T59328 CJYK13 117803656 IC50 = 5 nM T59328 C0MVG2 117803681 IC50 = 20 nM T59328 CXNZ08 117803686 IC50 = 14 nM T59328 CD93GO 117803687 IC50 = 5 nM T59328 CF7O9Z 117803889 IC50 = 9 nM T59328 CW6FL2 118073537 Ki = 9 nM T59328 CBV87I 118073538 Ki = 56 nM T59328 CKX0H7 118073560 IC50 = 1 nM T59328 CKRZ30 118073591 IC50 = 14 nM T59328 C42DMG 118073609 IC50 = 49 nM T59328 CID71C 118073630 IC50 = 194 nM T59328 CEDP63 118073633 IC50 = 6 nM T59328 C1U9WH 118073634 IC50 = 17 nM T59328 C2MDV0 118073642 IC50 = 3 nM T59328 C13PXJ 118073657 IC50 = 29 nM T59328 CGT4R5 118073677 Ki = 2 nM T59328 CMV6T3 118073685 Ki = 152 nM T59328 CKA98U 118073699 IC50 = 387 nM T59328 CUB7S0 118073727 Ki = 6 nM T59328 CLQO21 118073729 IC50 = 4 nM T59328 CVO01M 118073730 Ki = 36 nM T59328 C50FEY 118119835 IC50 = 60 nM T59328 CD8MX0 118223716 IC50 > 50000 nM T59328 CRM37Z 118223719 IC50 = 1.39 nM T59328 C5LNP8 118223723 IC50 > 50000 nM T59328 CB1I5P 118223929 IC50 > 50000 nM T59328 C52ETQ 118223987 IC50 = 16460 nM T59328 CEN18L 118224069 IC50 = 2.18 nM T59328 CTA5U1 118224099 IC50 < 2 nM T59328 CW72PI 118352095 IC50 = 218 nM T59328 CE4NX5 118352096 IC50 = 215 nM T59328 C93WJL 118352106 IC50 = 170 nM T59328 CBNZ41 118352115 IC50 = 80 nM T59328 C7QU3F 118352116 IC50 = 37 nM T59328 CDR52E 118352117 IC50 = 12 nM T59328 C7OUD9 118352135 IC50 = 101 nM T59328 CR7X3L 118352152 IC50 = 17 nM T59328 C2UYT6 118352158 IC50 > 1000 nM T59328 CDWL43 118352163 IC50 > 1000 nM T59328 C8U9AH 118352164 IC50 = 58 nM T59328 CMJ7F6 118352185 IC50 = 266 nM T59328 CQXJ61 118352193 IC50 = 48 nM T59328 CXH1G8 118352197 IC50 = 2 nM T59328 C5O8IG 118352198 IC50 = 192 nM T59328 CH8G4D 118352201 IC50 = 87 nM T59328 CVR8T2 118352210 IC50 = 45 nM T59328 CEM7X4 118352214 IC50 = 22 nM T59328 CC07LP 118352217 IC50 = 128 nM T59328 CAKI19 118514811 IC50 = 5.3 nM T59328 CIY3F2 118578874 IC50 = 287.4 nM T59328 CVHE23 118578939 IC50 = 6 nM T59328 C3D5UB 118661739 Ki = 57 nM T59328 C5Z6CQ 118661749 Ki = 1.1 nM T59328 C5B4MO 118661813 Ki = 34 nM T59328 C4P1SB 118662078 Ki = 44 nM T59328 C15RGE 118692362 IC50 = 20 nM T59328 CIU05O 118710979 IC50 = 10400 nM T59328 CJL49M 118710980 IC50 = 5400 nM T59328 C8WL4B 118710981 IC50 = 18300 nM T59328 C7WCP5 118710982 IC50 = 1100 nM T59328 C8PE2Y 118710983 IC50 = 4300 nM T59328 CBGV74 118710984 IC50 = 1300 nM T59328 CN38JS 118710985 IC50 = 8100 nM T59328 C51LZM 118710986 IC50 = 7000 nM T59328 CU3KJ9 118710987 IC50 = 200 nM T59328 C05DOU 118710988 IC50 = 16700 nM T59328 C4AHL2 118711367 IC50 > 10000 nM T59328 CW8JQ2 118712118 IC50 = 4800 nM T59328 CWO9B7 118715995 IC50 > 100000 nM T59328 C46QUT 118717614 IC50 = 77.2 nM T59328 CJC34Y 118717615 IC50 = 39.2 nM T59328 CFEP93 118717616 IC50 = 28.7 nM T59328 CEC4H0 118717617 IC50 = 89.6 nM T59328 CU2TG3 118717618 IC50 = 92.8 nM T59328 C5OL0W 118717619 IC50 = 110.2 nM T59328 CX0VC6 118719574 IC50 = 16000 nM T59328 C6EX4Q 118719575 IC50 = 6060000 nM T59328 CZEL74 118719576 IC50 = 57000 nM T59328 C01ZDF 118719577 IC50 = 66000 nM T59328 CK01PA 118719578 IC50 = 75000 nM T59328 C4NS1R 118719579 IC50 = 135000 nM T59328 CS3HJ5 118719580 IC50 = 9000000 nM T59328 C3L1TI 118720009 Ki = 28 nM T59328 CI5W9H 118720010 Ki = 14 nM T59328 COQ9S4 118720011 Ki = 18 nM T59328 CV4X8R 118720012 Ki = 114 nM T59328 C5FE8L 118720013 Ki = 423 nM T59328 C7T9VJ 118720014 Ki = 82 nM T59328 CGW7Z0 118721142 IC50 = 3.05 nM T59328 CZJB02 118721143 IC50 = 0.89 nM T59328 CO1B3H 118721144 IC50 = 0.47 nM T59328 C5IVR1 118721145 IC50 = 0.51 nM T59328 CYCQ59 118721146 IC50 = 0.32 nM T59328 CVL8Q3 118721147 IC50 = 0.66 nM T59328 C42NVI 118721148 IC50 = 1.08 nM T59328 C9MKR8 118721149 IC50 = 0.56 nM T59328 C0UA5Q 118721150 IC50 = 0.49 nM T59328 CJS7L9 118721151 IC50 = 0.5 nM T59328 CXHU43 118721152 IC50 = 38.3 nM T59328 CPL9H7 118721153 IC50 = 28.5 nM T59328 C29DWX 118721154 IC50 = 51.2 nM T59328 C9EJO7 118721155 IC50 = 15.1 nM T59328 CB8D5N 118721156 IC50 = 4.9 nM T59328 C5WFB8 118721157 IC50 = 3.43 nM T59328 C0S6RW 118721158 IC50 = 0.53 nM T59328 C20SQV 118721159 IC50 = 1.18 nM T59328 CB9SE1 118722338 IC50 = 2.6 nM T59328 C25AYC 118722339 IC50 = 2.55 nM T59328 CRIG46 118722340 IC50 = 37.9 nM T59328 CA5DI0 118722341 IC50 = 39.2 nM T59328 COB29E 118722342 IC50 = 9.5 nM T59328 CIH6Q8 118722343 IC50 = 11.2 nM T59328 CQ0IG7 118722344 IC50 = 5 nM T59328 C3KLI5 118723185 IC50 > 100000 nM T59328 CJX21C 118724340 IC50 = 0.77 nM T59328 C1C3WP 118724341 IC50 = 0.31 nM T59328 CZC2F3 118724342 IC50 = 0.52 nM T59328 CP9UL3 118724343 IC50 = 1.44 nM T59328 C7UX4R 118724344 IC50 = 0.32 nM T59328 C6Y3VE 118724345 IC50 = 0.65 nM T59328 CEF3I2 118724346 IC50 = 0.26 nM T59328 CW1E0M 118724347 IC50 = 0.57 nM T59328 CZ1G2X 118724348 IC50 = 0.54 nM T59328 CXD08A 118724349 IC50 = 30.5 nM T59328 C3J0KD 118724350 IC50 = 11.9 nM T59328 CY5X0E 118724351 IC50 = 16.6 nM T59328 CUT6Y3 118724352 IC50 = 35.5 nM T59328 CE6Q1K 118724353 IC50 = 20.1 nM T59328 C1J8EN 118724354 IC50 = 0.49 nM T59328 CB8MF7 118724355 IC50 = 0.37 nM T59328 CK28WP 118724356 IC50 = 0.33 nM T59328 CTSC96 118724357 IC50 = 0.78 nM T59328 CZ3LS6 118724358 IC50 = 0.82 nM T59328 C65JUN 118725950 IC50 = 8490 nM T59328 C9HWF5 118726554 IC50 = 1210 nM T59328 C9JKN5 118726555 IC50 = 950 nM T59328 CWYF91 118729842 IC50 = 162.3 nM T59328 CR54XL 118729843 IC50 = 90.3 nM T59328 CF3X9J 118729844 IC50 > 500 nM T59328 CT3Q6C 118729845 IC50 = 298.2 nM T59328 C1QWK6 118729846 IC50 = 226.4 nM T59328 CWUA61 118729847 IC50 = 306.6 nM T59328 C63CDP 118729848 IC50 = 103.2 nM T59328 C1WB7L 118729849 IC50 > 500 nM T59328 C8A7ZT 118729850 IC50 = 3.4 nM T59328 C9WDF4 118729851 IC50 = 102.2 nM T59328 CT08EZ 118729852 IC50 > 500 nM T59328 CG0C5B 118734111 IC50 = 153 nM T59328 COEJ71 118734112 IC50 = 53 nM T59328 CIEY96 118734113 IC50 = 23 nM T59328 CLN1C3 118734114 IC50 > 10000 nM T59328 C4U6AR 118734118 IC50 = 17 nM T59328 CV38ED 118734183 IC50 = 19 nM T59328 C1EI6R 118734184 IC50 = 629 nM T59328 CUJ3W6 118734185 IC50 = 8 nM T59328 CNDX69 118734186 IC50 = 23 nM T59328 CVPH90 118734187 IC50 = 27 nM T59328 CE8WN9 118734188 IC50 = 108 nM T59328 C9M7HI 118734189 IC50 = 275 nM T59328 C7LV4W 118734190 IC50 = 183 nM T59328 CF1ZN3 118734191 IC50 = 241 nM T59328 C7HA2M 118734192 IC50 > 10000 nM T59328 CXB50H 118734193 IC50 = 83 nM T59328 CKZG81 118734194 IC50 = 262 nM T59328 C0W8JD 118734195 IC50 > 10000 nM T59328 C8Y6UI 118734196 IC50 = 183 nM T59328 CMF34Q 118734200 IC50 = 150 nM T59328 CM1KO5 118734202 IC50 = 3883 nM T59328 CA2W7I 118734203 IC50 > 10000 nM T59328 CJ53YU 118734204 IC50 = 7904 nM T59328 C8Q5ZA 118734205 IC50 = 2079 nM T59328 CXW73G 118734207 IC50 = 1374 nM T59328 C6J8NH 118734208 IC50 = 415 nM T59328 C16HCZ 118734209 IC50 = 80 nM T59328 COI6J1 118734210 IC50 = 170 nM T59328 C45FIB 118734211 IC50 = 55 nM T59328 CLC85D 118734212 IC50 = 173 nM T59328 CC9S3Y 118734213 IC50 = 5 nM T59328 CG0JF1 118734214 IC50 = 18 nM T59328 CRQ98M 118734215 IC50 = 220 nM T59328 CY7ES4 118736528 IC50 = 7000 nM T59328 CT16XS 118736529 IC50 = 4800 nM T59328 CWNC90 118736530 IC50 > 10000 nM T59328 C8OP4R 118736531 IC50 > 10000 nM T59328 C75QPF 118736532 IC50 > 10000 nM T59328 CV9DL6 118736533 IC50 > 10000 nM T59328 C2VOS9 118736534 IC50 = 8700 nM T59328 CD4ZL0 118736535 IC50 > 10000 nM T59328 C18AYF 118736536 IC50 > 10000 nM T59328 CWI2O0 118736537 IC50 = 7200 nM T59328 C8HLE3 118736538 IC50 > 10000 nM T59328 CNTP03 118736539 IC50 > 10000 nM T59328 CYP1V5 118736540 IC50 > 10000 nM T59328 CMEK38 118736541 IC50 > 10000 nM T59328 C7EJ4B 118736542 IC50 > 10000 nM T59328 CU8D2K 118736543 IC50 > 10000 nM T59328 CAO94Z 118736544 IC50 = 3270 nM T59328 CCX29A 118736545 IC50 = 5600 nM T59328 CLI75H 118736546 IC50 > 10000 nM T59328 CQCX41 118737057 IC50 = 3518 nM T59328 CDBZ85 118738351 IC50 = 26 nM T59328 CJV62R 118738352 IC50 = 12.5 nM T59328 CSTB45 118738353 IC50 = 10.8 nM T59328 CM38XC 118738354 IC50 = 28 nM T59328 C1EDA6 118738355 IC50 = 59.9 nM T59328 C63SVY 118738356 IC50 = 11.4 nM T59328 CQ83JA 118738357 IC50 = 232.4 nM T59328 CUY8Z3 118900244 IC50 = 2.84 nM T59328 CB85RT 118900245 IC50 = 1.54 nM T59328 CR2X9A 118900269 IC50 = 153.5 nM T59328 CH3I9B 118900282 IC50 = 0.76 nM T59328 CI3TK4 118900289 IC50 = 1.48 nM T59328 C7V3DH 118900298 IC50 = 0.69 nM T59328 C0LIS1 118900305 IC50 = 0.94 nM T59328 CINT13 118900306 IC50 = 2.73 nM T59328 C9ARH1 118912888 IC50 = 6 nM T59328 CON03D 121231412 IC50 = 3 nM T59328 CBRZ51 121280156 IC50 > 600 nM T59328 CRQ3I6 121396150 IC50 = 11 nM T59328 CILM06 121423933 IC50 = 31 nM T59328 CN5CA4 121427628 IC50 = 5 nM T59328 CWA94G 122182409 IC50 > 100000 nM T59328 C02HIB 122186131 IC50 = 1100 nM T59328 C75JDA 122186132 IC50 = 100 nM T59328 CHG54X 122186133 IC50 > 10000 nM T59328 CS02EL 122186134 IC50 > 10000 nM T59328 CI35QX 122186135 IC50 = 400 nM T59328 C6PGI7 122186136 IC50 > 10000 nM T59328 CDKC89 122186137 IC50 = 300 nM T59328 CRH7T4 122186138 IC50 > 10000 nM T59328 CPO72V 122186139 IC50 = 2500 nM T59328 C56DAE 122186140 IC50 = 2100 nM T59328 CM5FZ6 122186141 Ki = 0.64 nM T59328 C98PCS 122186142 IC50 > 10000 nM T59328 C7R1JK 122186143 IC50 = 4900 nM T59328 CQCM53 122186144 IC50 = 1400 nM T59328 CS4LP5 122186145 IC50 = 900 nM T59328 C4VM5U 122186146 IC50 > 10000 nM T59328 C8VBX6 122186147 IC50 = 1900 nM T59328 CT9M5F 122186148 IC50 > 10000 nM T59328 CPD83K 122186149 IC50 = 1500 nM T59328 CA3SU2 122186150 Ki = 0.32 nM T59328 CI8RS6 122186151 IC50 = 8600 nM T59328 CU04WQ 122186152 IC50 = 700 nM T59328 C8DY3H 122186153 IC50 = 300 nM T59328 COMH39 122186154 IC50 = 3600 nM T59328 CTXU80 122186155 IC50 = 4900 nM T59328 C4P0JT 122188303 IC50 = 470 nM T59328 CSR50M 122188304 IC50 = 190 nM T59328 CRUV12 122188305 IC50 = 26 nM T59328 C6U3ER 122188306 IC50 = 5100 nM T59328 C3WB0T 122188307 IC50 > 10000 nM T59328 C3WLR4 122188308 IC50 > 10000 nM T59328 CMZX95 122188309 IC50 = 340 nM T59328 CC3BG6 122188310 IC50 > 10000 nM T59328 C57DPM 122188311 IC50 > 10000 nM T59328 C30MSH 122188312 IC50 = 560 nM T59328 C2F1DC 122188313 IC50 = 1300 nM T59328 CP8IB7 122188314 IC50 = 5500 nM T59328 C0C8EB 122188315 IC50 = 440 nM T59328 CEK54V 122188316 IC50 = 7800 nM T59328 C4S5QU 122188317 IC50 = 5700 nM T59328 C2H1AO 122188318 IC50 > 10000 nM T59328 C0VIM6 122188319 IC50 > 10000 nM T59328 C0D2EB 122188320 IC50 = 1200 nM T59328 C64GES 122188321 IC50 > 10000 nM T59328 C7GV9B 122188322 IC50 = 7500 nM T59328 C2LBT7 122188323 IC50 > 10000 nM T59328 C0ZIQ6 122188324 IC50 > 10000 nM T59328 CW3Q5T 122188325 IC50 > 10000 nM T59328 CKU2O7 122188326 IC50 > 10000 nM T59328 CS3Z2X 122188327 IC50 = 780 nM T59328 CFO57L 122188328 IC50 > 10000 nM T59328 CNF7Q2 122188329 IC50 = 7.3 nM T59328 C7RU0L 122188330 IC50 > 10000 nM T59328 CGZJ16 122188331 IC50 > 10000 nM T59328 C8O7SU 122188332 IC50 = 130 nM T59328 C8G4QO 122188333 IC50 = 2300 nM T59328 CO96BU 122188334 IC50 = 140 nM T59328 C0HBC8 122188335 IC50 = 53 nM T59328 C79UWR 122188336 IC50 = 20 nM T59328 CCP8B1 122188337 IC50 = 8.7 nM T59328 C4BOF5 122188338 IC50 = 160 nM T59328 CAS18Q 122188339 IC50 > 10000 nM T59328 CYPA94 122188340 IC50 > 10000 nM T59328 C52ERC 122188341 IC50 = 660 nM T59328 CYW1M5 122188342 IC50 = 1500 nM T59328 CCV6T9 122189237 IC50 = 5283 nM T59328 C61RXE 122189241 IC50 = 4824 nM T59328 CG7P6E 122189248 IC50 = 0.037 nM T59328 C0YZ4K 122191926 IC50 > 1000 nM T59328 C6Q5CB 122191927 IC50 = 1.2 nM T59328 CZG10A 122191928 IC50 = 573.6 nM T59328 CB9XO4 122191929 IC50 = 102.3 nM T59328 C7R8AM 122191930 IC50 > 1000 nM T59328 C2GP3K 122191931 IC50 = 5.4 nM T59328 CH0J8K 122191932 IC50 = 1.2 nM T59328 CM8G5F 122191933 IC50 = 3 nM T59328 CZB2R1 122191934 IC50 = 510.2 nM T59328 CO43WT 122191935 IC50 = 133.9 nM T59328 CB3FU0 122191936 IC50 = 9 nM T59328 CVEQ28 122191937 IC50 > 1000 nM T59328 C8YIT6 122191938 IC50 = 147.4 nM T59328 C31QLD 122191939 IC50 = 26.9 nM T59328 C1JQ0L 122191940 IC50 = 8.9 nM T59328 C6CGK1 122191941 IC50 = 5.5 nM T59328 C0SAT2 122191942 IC50 > 1000 nM T59328 C4M3OA 122191943 IC50 > 1000 nM T59328 CB8DC6 122191944 IC50 > 1000 nM T59328 CZFO12 122191945 IC50 > 1000 nM T59328 C7YZE5 122191946 IC50 > 1000 nM T59328 C7NV0K 122191947 IC50 > 1000 nM T59328 CPK50T 122191948 IC50 = 0.9 nM T59328 CF4E8L 122191949 IC50 = 2.1 nM T59328 CTI7K9 122191950 IC50 = 6.5 nM T59328 C83TUO 122191951 IC50 = 9.6 nM T59328 CFS29N 122191952 IC50 = 6.9 nM T59328 C25QVG 122191953 IC50 = 141 nM T59328 C5O8VS 122191954 IC50 = 7 nM T59328 CY24OJ 122191955 IC50 = 5.3 nM T59328 C2A9MG 122191956 IC50 = 3.3 nM T59328 CVT7W4 122191957 IC50 = 2.4 nM T59328 CRM0T2 122191958 IC50 = 5.6 nM T59328 C8ZPL5 122191959 IC50 = 7.9 nM T59328 CNU1X5 122191960 IC50 = 4.2 nM T59328 CL8M2N 122191961 IC50 = 6.4 nM T59328 C4X7SD 122192466 IC50 > 10000 nM T59328 CJ6RO8 122193596 IC50 > 10000 nM T59328 CB6M4T 122193759 IC50 > 10000 nM T59328 C65XUZ 122193760 IC50 > 10000 nM T59328 CHF47Y 122193761 IC50 > 10000 nM T59328 C1XHI4 122193762 IC50 = 7710 nM T59328 CNX0Q2 122193763 IC50 > 10000 nM T59328 CWV0C3 122193764 IC50 > 10000 nM T59328 CSG98Y 122193765 IC50 = 3950 nM T59328 C1SED2 122193766 IC50 > 10000 nM T59328 CINA05 122193767 IC50 > 10000 nM T59328 C27WGV 122193768 IC50 > 10000 nM T59328 CCLQ75 122193769 IC50 > 10000 nM T59328 CXDR48 122193770 IC50 > 10000 nM T59328 C96LDU 122193771 IC50 > 10000 nM T59328 C50HEA 122193772 IC50 > 10000 nM T59328 CPA8C5 122193773 IC50 > 10000 nM T59328 C83XVM 122193778 IC50 = 21180 nM T59328 CIS0B2 122193779 IC50 = 21560 nM T59328 C26POY 122193780 IC50 = 45700 nM T59328 C59RDU 122193840 IC50 = 3290 nM T59328 CXE87R 122193841 IC50 = 1260 nM T59328 CM8N1W 122195059 IC50 = 348 nM T59328 CC5KB6 122195541 IC50 = 4 nM T59328 CKG14J 122195542 IC50 = 543 nM T59328 CIPZ05 122195677 IC50 = 186 nM T59328 C4V5WK 122195678 IC50 = 29 nM T59328 C03XJB 122195679 IC50 > 10000 nM T59328 C2CM8S 122195680 IC50 = 35 nM T59328 CIC6N1 122195681 IC50 = 227 nM T59328 C3F1YP 122195682 IC50 = 23 nM T59328 C4IMA2 122195683 IC50 > 10000 nM T59328 C8TK1W 122195684 IC50 = 812 nM T59328 C4FXV5 122195685 IC50 = 1020 nM T59328 C47QYW 122195686 IC50 > 10000 nM T59328 CZC4K1 122195687 IC50 = 445 nM T59328 CK0Q3A 122195688 IC50 = 3050 nM T59328 CLTG90 122195689 IC50 = 9 nM T59328 C0TX3A 122195690 IC50 = 31 nM T59328 C52BMS 122195691 IC50 = 1460 nM T59328 C1KXL8 122205446 IC50 = 280 nM T59328 C4XIQ7 122205447 IC50 = 21 nM T59328 C3BL8I 122205448 IC50 > 1000 nM T59328 C37ICD 122417697 IC50 = 363.3 nM T59328 C9D5RK 122417700 IC50 = 57.8 nM T59328 CQD76R 122417702 IC50 = 76.1 nM T59328 C47VHI 122417706 IC50 = 6.7 nM T59328 CBF3G5 122417707 IC50 = 10.9 nM T59328 C69PHO 122417709 IC50 = 3.6 nM T59328 CW64ZC 122417712 IC50 = 53.1 nM T59328 C5BMI1 122417713 IC50 > 1000 nM T59328 C1YRN4 122417718 IC50 = 82.5 nM T59328 CE45KB 122417721 IC50 = 416.1 nM T59328 C9LK2Y 122417722 IC50 > 1000 nM T59328 C5RD4P 122417724 IC50 = 232.3 nM T59328 CAG29M 122417725 IC50 = 351.8 nM T59328 C6QMU4 122417730 IC50 = 16.7 nM T59328 C90XRZ 122417735 IC50 = 8.1 nM T59328 CFSK74 122417740 IC50 > 1000 nM T59328 CWT4F3 122417747 IC50 = 102.6 nM T59328 CHY1Z0 122417753 IC50 > 1000 nM T59328 CC04MJ 122417757 IC50 = 46.28 nM T59328 C35XVJ 122417762 IC50 = 43.8 nM T59328 C9WJ6T 122417763 IC50 = 36.2 nM T59328 C19SAP 122417767 IC50 = 9.2 nM T59328 C1VP7E 122417768 IC50 = 22.5 nM T59328 CV68FJ 122417770 IC50 = 27.3 nM T59328 CIG7Y6 122417773 IC50 > 1000 nM T59328 CD37VR 122417777 IC50 = 10.5 nM T59328 C0IJR1 122417781 IC50 = 4.4 nM T59328 C0XFJ2 122417784 IC50 = 24.1 nM T59328 C4LV6K 122417787 IC50 = 162.7 nM T59328 C2VP7F 122417788 IC50 = 139 nM T59328 C8UF2Q 122417837 IC50 = 184.5 nM T59328 C6DAO2 122417839 IC50 = 313.6 nM T59328 CDT5O1 122417840 IC50 = 23.7 nM T59328 CJ6D9N 122417841 IC50 = 74.6 nM T59328 CAM13U 122417842 IC50 = 387.8 nM T59328 CFL0M8 122417848 IC50 > 1000 nM T59328 C1TIR7 122417852 IC50 = 247.2 nM T59328 CWL2N6 122417856 IC50 = 109.1 nM T59328 C9VTO7 122417858 IC50 = 2 nM T59328 C9QB1R 122417864 IC50 = 9.7 nM T59328 C6QHB4 122484585 IC50 = 0.3 nM T59328 CRT93E 122484586 IC50 = 1.2 nM T59328 CF7ME6 122484587 IC50 = 16 nM T59328 CX8EC3 122484589 IC50 = 111 nM T59328 C2E8NC 122484594 IC50 = 14 nM T59328 CJ63LF 122484678 IC50 = 70 nM T59328 C6DP2N 122484680 IC50 = 68 nM T59328 C2SXK9 122484682 IC50 = 314 nM T59328 C8MJ4P 122484684 IC50 = 180 nM T59328 C1U2WJ 122484694 IC50 = 0.4 nM T59328 CJC73G 122484695 IC50 = 3.8 nM T59328 C4AUD3 122484700 IC50 = 0.8 nM T59328 CS58YZ 122484702 IC50 = 30 nM T59328 CX6KW7 122484733 IC50 = 115 nM T59328 CV63PN 122484734 IC50 = 1 nM T59328 C1NPL5 122484735 IC50 = 6.8 nM T59328 C01SPL 122484737 IC50 = 0.7 nM T59328 CLM7K3 122604539 IC50 > 10000 nM T59328 C01JHI 122604566 IC50 > 10000 nM T59328 CIR1B3 123134714 IC50 = 2.4 nM T59328 CY30FL 123752658 IC50 > 100 nM T59328 CZAY93 124197376 IC50 = 4.1 nM T59328 C5T9NG 124197380 IC50 = 5 nM T59328 CZFG57 124197588 IC50 = 8.4 nM T59328 CH0B7X 124222449 Ki = 161 nM T59328 CIP4Q6 124435382 IC50 = 147 nM T59328 CAXY02 125461985 IC50 = 2 nM T59328 CCX79B 126667178 IC50 = 2100 nM T59328 C97OIS 127024859 IC50 = 21 nM T59328 CBU92A 127024861 IC50 = 7 nM T59328 CJB02T 127024862 IC50 = 0.5 nM T59328 C5P6VB 127024863 IC50 = 4 nM T59328 CEI65V 127024864 IC50 = 0.4 nM T59328 CIB0W9 127024865 IC50 = 3 nM T59328 CE89QB 127024882 IC50 > 10000 nM T59328 CUF81C 127025156 IC50 > 500 nM T59328 CP3LK5 127025157 IC50 = 14.83 nM T59328 C8QKX6 127025158 IC50 = 97.22 nM T59328 C86RIQ 127025203 IC50 = 300 nM T59328 CDQ52G 127025443 IC50 = 48.81 nM T59328 CZH1K2 127025487 Ki > 2000 nM T59328 COA80E 127025789 IC50 = 2 nM T59328 CL4YH3 127025790 IC50 = 0.9 nM T59328 CYQ2U3 127025791 IC50 = 2 nM T59328 CZRI81 127025792 IC50 = 21 nM T59328 C8KXV1 127025843 IC50 > 1000 nM T59328 CG3T9I 127026061 IC50 = 6 nM T59328 CVYD73 127026080 IC50 = 0.9 nM T59328 C27YJQ 127026081 IC50 = 2 nM T59328 CFV5O3 127026082 IC50 = 1.5 nM T59328 CGT0I1 127026385 Ki = 10.4 nM T59328 CQ8EW1 127026406 IC50 = 9 nM T59328 CW6PB1 127026407 IC50 = 3 nM T59328 CVRP85 127026408 IC50 = 20 nM T59328 C3Y0XF 127026464 IC50 = 5 nM T59328 C1V2ZA 127026465 IC50 = 19 nM T59328 C7A4QX 127026466 IC50 = 7 nM T59328 CCI6J7 127026467 IC50 = 41 nM T59328 CEM1T3 127026690 IC50 = 276 nM T59328 CI3HN6 127026710 IC50 = 0.5 nM T59328 CY1K9D 127027073 IC50 = 48 nM T59328 C41EAT 127027074 IC50 = 5 nM T59328 CBA80X 127027086 IC50 = 13 nM T59328 CWK63L 127027087 IC50 = 59 nM T59328 CRQ0E7 127027088 IC50 = 8 nM T59328 CV34HC 127027089 IC50 = 5 nM T59328 CIKQ57 127027090 IC50 = 26 nM T59328 CBT52X 127027296 IC50 = 66.59 nM T59328 CS6TJ8 127027297 IC50 = 90.57 nM T59328 C0EZA2 127027298 IC50 > 500 nM T59328 CER0Q3 127027305 IC50 = 78.17 nM T59328 CAH9J6 127027306 IC50 = 476.66 nM T59328 CN3SW5 127027307 IC50 = 71.82 nM T59328 CC0R4L 127027308 IC50 = 121.09 nM T59328 C9E7CQ 127027332 IC50 > 10000 nM T59328 CA59WC 127027333 IC50 = 730 nM T59328 CQXW85 127027334 IC50 > 10000 nM T59328 CPLE01 127027335 IC50 > 10000 nM T59328 CSM76Y 127027336 IC50 > 10000 nM T59328 C7EYC2 127027620 IC50 = 26.56 nM T59328 C12ODR 127027621 IC50 = 131.09 nM T59328 CA7JW5 127027622 IC50 = 455.17 nM T59328 CMT3C7 127027623 IC50 = 290.46 nM T59328 C0T3HO 127027641 IC50 = 495.3 nM T59328 CLO6P4 127027642 IC50 = 165.6 nM T59328 C14WBS 127027666 IC50 = 8 nM T59328 CUG53Q 127027694 Ki = 0.6 nM T59328 CE1BH6 127027695 Ki = 844 nM T59328 CM2S6K 127027696 Ki = 389 nM T59328 CRZA23 127027741 IC50 = 159 nM T59328 CV7R6H 127027985 IC50 = 2 nM T59328 C0Q6RG 127027992 IC50 = 130 nM T59328 CO3P6I 127028013 Ki > 2000 nM T59328 C3O4AR 127028014 Ki = 3 nM T59328 C1A3FO 127028015 Ki = 2 nM T59328 CG7ZB1 127028016 Ki = 8 nM T59328 CW5EY8 127028017 Ki = 17 nM T59328 CE62DA 127028049 IC50 = 4.52 nM T59328 C0HAR2 127028050 IC50 = 2.92 nM T59328 C82RGS 127028051 IC50 = 10.8 nM T59328 C7SIV9 127028052 IC50 = 5.01 nM T59328 CH1TO3 127028299 Ki = 134 nM T59328 C04MHS 127028310 IC50 = 150 nM T59328 C85ZEY 127028311 IC50 = 20 nM T59328 C5V3SU 127028312 IC50 = 1330 nM T59328 C6C0QK 127028313 IC50 = 690 nM T59328 CXE58H 127028337 Ki = 17 nM T59328 CZK9V1 127028338 Ki = 747 nM T59328 CG7I9K 127028339 Ki > 2000 nM T59328 CIZ7M1 127028340 Ki > 2000 nM T59328 C43XYB 127028671 Ki = 22.4 nM T59328 CG9M4V 127028672 Ki = 4 nM T59328 CI7TC8 127028673 Ki = 16 nM T59328 CR9A4B 127028681 Ki = 57 nM T59328 CK71GH 127028959 Ki = 6.5 nM T59328 C9XH6D 127028969 IC50 = 1110 nM T59328 C9CMQ6 127028970 IC50 = 4610 nM T59328 CXFB96 127028971 IC50 > 10000 nM T59328 CYAT13 127028990 Ki = 519 nM T59328 C4QX6U 127028991 Ki = 85 nM T59328 CVR5S1 127028992 Ki = 104 nM T59328 C4Y8CR 127028993 Ki = 732 nM T59328 CFN3D7 127028994 Ki = 5.6 nM T59328 CLK2Z3 127028995 Ki = 175 nM T59328 C64UOV 127029263 IC50 = 760 nM T59328 C69BON 127029520 IC50 = 13 nM T59328 C1XD6R 127029809 IC50 > 100000 nM T59328 CI1E5W 127029864 IC50 = 582.17 nM T59328 C9CDQ5 127029901 IC50 = 434.1 nM T59328 C4I7ZN 127029902 IC50 = 353.7 nM T59328 CHPZ40 127029903 IC50 = 823.9 nM T59328 C4KF0T 127030085 Ki = 15 nM T59328 CG2DM3 127030086 Ki = 32 nM T59328 CTA3J6 127030119 Ki = 346 nM T59328 CO0I4A 127030120 Ki = 82 nM T59328 C4WY3P 127030121 Ki = 155 nM T59328 C6PK2L 127030122 Ki = 629 nM T59328 CVBF01 127030212 IC50 > 10000 nM T59328 CI93ZA 127030213 IC50 > 10000 nM T59328 C70DZQ 127030241 IC50 = 594.5 nM T59328 C1D8OL 127030242 IC50 = 518.6 nM T59328 C60QMN 127030384 Ki = 10 nM T59328 C8LQV4 127030516 IC50 > 10000 nM T59328 CV2EA7 127030757 Ki > 2060 nM T59328 CT7SX1 127031071 Ki = 108 nM T59328 C4U1NV 127031072 Ki = 95 nM T59328 CD4RB2 127031073 Ki = 145 nM T59328 CL31XR 127031074 Ki > 688 nM T59328 C0BR2L 127031164 IC50 = 89.6 nM T59328 CN9IV4 127031165 IC50 = 186.9 nM T59328 C2O1VX 127031166 IC50 = 829.2 nM T59328 CS12RU 127031435 IC50 > 10000 nM T59328 CZXP62 127031750 IC50 > 10000 nM T59328 CD45KQ 127031941 Ki = 61 nM T59328 C3E5YO 127032014 IC50 > 10000 nM T59328 C2ZD8S 127032024 IC50 > 10000 nM T59328 CXWY73 127032324 IC50 > 10000 nM T59328 C42UOD 127032352 IC50 = 245.1 nM T59328 CV42MI 127032353 IC50 = 63.1 nM T59328 CJ59GA 127032541 Ki = 330 nM T59328 CS40XR 127032999 IC50 = 137.9 nM T59328 CQ1I3B 127033227 Ki = 37 nM T59328 C59MVH 127033228 Ki > 2060 nM T59328 CR2P3O 127033504 Ki = 51 nM T59328 CB35SE 127033505 Ki = 15 nM T59328 C2GLU3 127033506 Ki = 12 nM T59328 C81SKW 127033507 Ki = 78 nM T59328 C46AWH 127033508 Ki = 26 nM T59328 CWIO91 127033509 Ki = 31 nM T59328 CJZT54 127033800 Ki = 625 nM T59328 CL7P4Q 127033902 Ki = 590 nM T59328 C9BYR7 127034155 IC50 = 460 nM T59328 CL67CH 127034156 IC50 = 115.9 nM T59328 C3ZTY9 127034157 IC50 = 99 nM T59328 C5EM4W 127034158 IC50 = 456.2 nM T59328 C97FGP 127034305 Ki = 349 nM T59328 C52FRX 127034424 IC50 = 211.4 nM T59328 CEDK31 127034582 Ki = 144 nM T59328 CKS28E 127034802 IC50 = 350 nM T59328 CWRB15 127034986 IC50 = 71.71 nM T59328 CM09WL 127035009 IC50 = 18.04 nM T59328 CDU87A 127035163 IC50 = 94.82 nM T59328 CPN2Q6 127035597 Ki = 196 nM T59328 CEPL09 127036182 IC50 = 310.76 nM T59328 C87BIU 127036183 IC50 = 102.93 nM T59328 CR0NI6 127036477 IC50 = 317.12 nM T59328 CM17TO 127036596 IC50 = 24.81 nM T59328 C3SPE9 127036731 Ki = 7.4 nM T59328 CGOK31 127036732 Ki = 9.5 nM T59328 C52JBY 127036758 IC50 = 362 nM T59328 C72EXH 127036764 IC50 = 189.49 nM T59328 CKX40V 127037812 IC50 > 10000 nM T59328 C93RQT 127038361 IC50 = 9190 nM T59328 CHMT84 127038362 IC50 = 4480 nM T59328 CVU8Z4 127038363 IC50 = 3220 nM T59328 CB73NS 127038364 IC50 = 7880 nM T59328 C70RUP 127038480 IC50 > 10000 nM T59328 CEG89U 127038628 IC50 = 25580 nM T59328 CJHQ62 127038729 IC50 = 3200 nM T59328 CSV0T8 127039237 IC50 = 9.1 nM T59328 C18SAK 127039275 IC50 = 4130 nM T59328 C5GJ1F 127039276 IC50 = 5960 nM T59328 CYNR48 127039277 IC50 = 301.3 nM T59328 CLI54D 127039495 IC50 = 1680 nM T59328 C03PVF 127039496 IC50 = 2270 nM T59328 CRS60P 127039497 IC50 = 5670 nM T59328 C4BY1V 127039518 IC50 = 11570 nM T59328 C87AFX 127039599 IC50 = 6683.44 nM T59328 CUVR09 127039608 IC50 = 8540 nM T59328 COE17A 127039609 IC50 = 21310 nM T59328 C93XHQ 127039610 IC50 = 9594.01 nM T59328 CXLQ81 127039662 IC50 = 12240 nM T59328 CW4S0U 127039718 IC50 = 3890 nM T59328 C8BSO6 127039719 IC50 = 5430 nM T59328 CNH94T 127039720 IC50 = 2550 nM T59328 C01LGZ 127039804 IC50 = 4670 nM T59328 CO4N6V 127039812 IC50 = 790 nM T59328 CEU27C 127039813 IC50 = 2350 nM T59328 C48BVH 127039814 IC50 = 720 nM T59328 CBM41V 127039833 IC50 = 790 nM T59328 C91FAK 127039834 IC50 = 680 nM T59328 C6OU4T 127039835 IC50 = 2520 nM T59328 C3N2YV 127039870 IC50 = 3.6 nM T59328 CKT2I9 127039915 IC50 = 26920 nM T59328 CEQA86 127039935 IC50 = 600 nM T59328 CTK6W3 127039936 IC50 = 1450 nM T59328 CB3X9Y 127039944 IC50 = 15160 nM T59328 CAL3D1 127039945 IC50 = 7379.04 nM T59328 CB5KT1 127039946 IC50 = 9260 nM T59328 C03XGE 127040180 IC50 = 2380 nM T59328 C7CNB9 127040181 IC50 = 4320 nM T59328 C8PK1U 127040288 IC50 = 5023.43 nM T59328 CT4U6D 127040940 IC50 = 6580 nM T59328 CJ8E7C 127040941 IC50 = 1260 nM T59328 CA6RH0 127040942 IC50 = 10690 nM T59328 CP6D1T 127040943 IC50 = 10939.56 nM T59328 CYM0T6 127041396 IC50 = 3560 nM T59328 CXM5Q6 127041397 IC50 = 4490 nM T59328 CJI9D7 127041398 IC50 = 3780 nM T59328 CGX1C5 127041399 IC50 = 2560 nM T59328 C6Z5KQ 127041488 IC50 = 860 nM T59328 C3WCN8 127041777 IC50 > 10000 nM T59328 CV53TB 127041787 IC50 = 1510 nM T59328 CP03MA 127042285 IC50 = 1.12 nM T59328 C4M7QX 127042286 IC50 = 15.4 nM T59328 CK5H8B 127042641 IC50 = 2.01 nM T59328 CNA9F0 127042642 IC50 = 4.62 nM T59328 CQNL56 127042643 IC50 = 4.71 nM T59328 C5PFK0 127042644 IC50 = 6.02 nM T59328 C1G9QI 127042685 IC50 = 2890 nM T59328 CZ3J4V 127042686 IC50 = 3670 nM T59328 C27XTM 127042687 IC50 = 5100 nM T59328 CUY35P 127042939 IC50 = 1.63 nM T59328 CP15ZX 127043295 IC50 = 2.97 nM T59328 C1ID2U 127044206 IC50 = 880 nM T59328 CV0F3N 127045112 IC50 = 28.2 nM T59328 CTPY32 127045266 IC50 = 44.1 nM T59328 CWI8Q2 127045267 IC50 = 3.58 nM T59328 CV5I8S 127045270 IC50 = 31.9 nM T59328 CL9BQ0 127045740 IC50 = 4.4 nM T59328 CG1OT5 127045741 IC50 = 38.8 nM T59328 C3M7AZ 127045742 IC50 = 3.7 nM T59328 CHK16Q 127045929 IC50 > 1000 nM T59328 CG70DF 127046321 IC50 = 0.4 nM T59328 CHT3M0 127046322 IC50 = 0.7 nM T59328 C3R7UG 127046487 IC50 = 7.3 nM T59328 CRWO38 127046488 IC50 = 1.8 nM T59328 CAK4O6 127046533 IC50 = 3.6 nM T59328 CZ6A2F 127046534 IC50 = 5.8 nM T59328 CO4N3J 127047042 IC50 = 49000 nM T59328 CL18YE 127047185 IC50 = 34000 nM T59328 C8TIY1 127047186 IC50 = 35000 nM T59328 CVC5W1 127047187 IC50 = 15000 nM T59328 CW5X1G 127047188 IC50 = 38000 nM T59328 CO96WN 127047445 IC50 = 9.6 nM T59328 CY3J0C 127047591 IC50 > 1000 nM T59328 C81WZQ 127048296 IC50 = 259 nM T59328 CDL7Z4 127048297 IC50 > 500 nM T59328 CGXU78 127048860 IC50 = 20.5 nM T59328 C7Q0FC 127048861 IC50 = 58.8 nM T59328 C0V7YZ 127048976 IC50 = 2.04 nM T59328 CMTG09 127048977 IC50 = 0.854 nM T59328 CDWM04 127048978 IC50 = 0.662 nM T59328 CPH4B3 127048979 IC50 = 3.96 nM T59328 CN1WT6 127048980 IC50 = 1.43 nM T59328 CQ83OB 127048981 IC50 = 0.772 nM T59328 CAY75H 127048991 EC50 = 360 nM T59328 C8M1LU 127049195 IC50 = 25.86 nM T59328 C4X2CJ 127049305 EC50 = 1780 nM T59328 CVZE82 127049306 EC50 = 18 nM T59328 C5ZF0X 127049307 EC50 = 150 nM T59328 CAX68G 127049308 EC50 = 10 nM T59328 CR64FG 127049380 IC50 = 1.34 nM T59328 CLF41Y 127049383 IC50 = 5.52 nM T59328 CVH72U 127049689 IC50 = 0.803 nM T59328 CP2NO1 127049690 IC50 = 194 nM T59328 C6A2IV 127050067 IC50 = 1.98 nM T59328 C1TAI8 127050068 IC50 = 294.6 nM T59328 CIV53M 127050256 EC50 = 22 nM T59328 C82WZB 127050549 EC50 = 1340 nM T59328 C16LRJ 127050550 EC50 = 390 nM T59328 CR3KX5 127050551 EC50 > 20000 nM T59328 C95CNQ 127050554 IC50 = 5.06 nM T59328 C1PFS7 127050555 IC50 = 247 nM T59328 CJ5L8A 127050556 IC50 < 0.495 nM T59328 CB3G8V 127050557 IC50 = 1.5 nM T59328 CYT6X9 127050558 EC50 = 24 nM T59328 C1PHY6 127050559 EC50 = 15 nM T59328 C8I2MC 127050881 EC50 = 550 nM T59328 CJ4WY0 127050882 EC50 = 7 nM T59328 CBS36H 127051046 IC50 = 200.3 nM T59328 CE7B3D 127051146 IC50 = 200 nM T59328 C6XHP2 127051445 IC50 < 1 nM T59328 CO29UV 127051446 EC50 > 30000 nM T59328 CQW87Z 127051447 EC50 = 73 nM T59328 CX31ZJ 127051448 EC50 = 23 nM T59328 CD0CG5 127051556 IC50 = 25.53 nM T59328 CHF7B5 127051692 IC50 = 9040 nM T59328 C4KLU2 127051866 IC50 = 4.54 nM T59328 CI9Y4N 127051867 IC50 = 1.19 nM T59328 CH4AJ8 127052082 EC50 = 14900 nM T59328 C7V9BT 127052091 IC50 = 2.25 nM T59328 CHQG07 127052092 IC50 = 80 nM T59328 C9XM4K 127052093 IC50 = 2.26 nM T59328 CSO2J4 127052094 EC50 = 12 nM T59328 C1AK9H 127052095 EC50 = 24 nM T59328 CQG69I 127052096 EC50 = 15 nM T59328 CH51IT 127052097 EC50 = 9 nM T59328 C5N0QK 127052408 IC50 = 296 nM T59328 CO3E8G 127052409 IC50 = 9.05 nM T59328 CB5YE2 127052414 EC50 = 14 nM T59328 CZ52FH 127052605 IC50 = 18.48 nM T59328 C0D6UI 127052606 IC50 = 21.95 nM T59328 CSM21N 127052640 IC50 = 192000 nM T59328 CN6V5E 127052874 IC50 > 300000 nM T59328 C1T8EL 127052875 IC50 > 300000 nM T59328 CUO7X0 127052876 IC50 = 7920 nM T59328 CGKZ89 127052877 IC50 = 81200 nM T59328 C1PK0X 127052898 IC50 = 83.88 nM T59328 CZ37CP 127052899 IC50 = 97.18 nM T59328 CNGZ92 127052993 IC50 = 2.92 nM T59328 CBHF87 127052994 IC50 = 62 nM T59328 CS5T2B 127053079 IC50 = 37.81 nM T59328 CIU72D 127264586 IC50 = 5.3 nM T59328 C8ZM1T 129281909 IC50 = 3.6 nM T59328 C2LWZ1 129318964 IC50 > 10000 nM T59328 C0XS4M 129896681 IC50 > 10000 nM T59328 C0FM1R 130196825 IC50 = 1970 nM T59328 CGOQ27 130412632 IC50 = 1.6 nM T59328 CFA3V6 132020316 IC50 = 73.1 nM T59328 CUO0C5 132156633 IC50 > 10000 nM T59328 CV8DP9 132487332 IC50 = 3.23 nM T59328 C0G9TV 132495274 IC50 = 0.12 nM T59328 C51EID 132496692 IC50 < 0.5 nM T59328 C0V2WX 132578497 IC50 = 3.3 nM T59328 CRV07S 132597737 IC50 = 0.3 nM T59328 CL6E4J 132601725 IC50 > 25000 nM T59328 C53OJM 132607333 IC50 = 980.83 nM T59328 CA6TN4 132609257 IC50 = 6.4 nM T59328 CMI3Q0 132819888 IC50 = 690 nM T59328 CERS64 132937256 IC50 > 30000 nM T59328 C46ORZ 132938092 IC50 = 21 nM T59328 C32QRI 132938093 IC50 = 11 nM T59328 CN9SD7 132942957 IC50 = 92.5 nM T59328 CMP2S9 132942958 IC50 = 7.2 nM T59328 CDMF97 134130282 IC50 > 150000 nM T59328 C2H6PW 134130554 IC50 > 150000 nM T59328 CM5T6K 134130825 IC50 = 8 nM T59328 CWF16B 134131331 IC50 > 100000 nM T59328 CLV5I3 134131586 IC50 > 150000 nM T59328 C79SPC 134131685 IC50 = 5200 nM T59328 CC1EB5 134131929 IC50 = 4 nM T59328 CTC7P8 134132114 IC50 = 11 nM T59328 CHW59N 134132187 IC50 = 240 nM T59328 CE1Y8U 134132335 IC50 = 280 nM T59328 CA7J2D 134132574 IC50 = 4.2 nM T59328 C6CYV4 134132651 IC50 > 10000 nM T59328 C3NEU6 134133052 IC50 = 86 nM T59328 CS79UR 134133060 IC50 = 460 nM T59328 C1BTI2 134133235 IC50 = 5.4 nM T59328 CMZG34 134133313 IC50 = 8 nM T59328 C1VOY4 134133329 IC50 = 8 nM T59328 C6IU4F 134133491 IC50 = 500 nM T59328 CZT6O0 134133815 IC50 = 4.6 nM T59328 CI53QU 134133842 IC50 = 64 nM T59328 CG8M5O 134134176 IC50 = 130 nM T59328 CX2WN6 134134364 IC50 = 16 nM T59328 CTZ84R 134134811 IC50 = 4700 nM T59328 C15PJY 134134898 IC50 = 0.4 nM T59328 CH3QN8 134135021 IC50 = 5.6 nM T59328 CPJG85 134135151 IC50 = 601 nM T59328 C3COF8 134135258 IC50 = 4.4 nM T59328 CSZX25 134135323 IC50 = 16 nM T59328 CR5F3L 134135362 IC50 = 668 nM T59328 CDMJ75 134135414 IC50 = 3.6 nM T59328 CV4Q0M 134135529 IC50 = 763 nM T59328 CEQ1M7 134135734 IC50 = 235 nM T59328 CF9NZ6 134135902 IC50 = 118.7 nM T59328 CUL3Q0 134136044 IC50 = 300 nM T59328 C1GVQ7 134136098 IC50 = 175 nM T59328 C3G7TQ 134136245 IC50 = 36 nM T59328 CUP13V 134136269 IC50 = 0.6 nM T59328 CD1O7N 134136322 IC50 = 4649 nM T59328 CZD0J5 134136450 IC50 = 8500 nM T59328 C3LX0Z 134136666 IC50 = 47 nM T59328 C9FZ3A 134136788 IC50 = 587 nM T59328 CL4PT1 134137211 IC50 > 10000 nM T59328 CG92RQ 134137314 IC50 = 593 nM T59328 CYGZ85 134137500 IC50 = 10 nM T59328 CN79XJ 134137614 IC50 = 78 nM T59328 C1U2MV 134137679 IC50 = 460 nM T59328 CJC1E8 134137789 IC50 = 6.4 nM T59328 CK15UI 134137837 IC50 = 502 nM T59328 CJ7C1N 134137974 IC50 = 14 nM T59328 C2L8OB 134138134 IC50 = 510 nM T59328 CC86FV 134138222 IC50 = 136 nM T59328 C3RA6C 134138227 IC50 = 0.27 nM T59328 C5JH9E 134138228 IC50 = 29 nM T59328 CY3U6V 134138310 IC50 = 36 nM T59328 CTY21M 134138472 IC50 = 98.2 nM T59328 CC42DJ 134138534 IC50 = 22 nM T59328 C4QSZ5 134138566 IC50 = 29 nM T59328 CZU97C 134138682 IC50 = 2 nM T59328 C0GT4V 134138751 IC50 = 9 nM T59328 CLG84S 134138800 IC50 = 5.3 nM T59328 C6RGN8 134138812 IC50 = 30 nM T59328 C58FUC 134139047 IC50 = 2 nM T59328 C45HRS 134139393 IC50 = 194 nM T59328 CG91IQ 134139430 IC50 = 79 nM T59328 C5OEI3 134139438 IC50 = 23 nM T59328 C6U5WE 134139490 IC50 = 94 nM T59328 CA7PD8 134139534 IC50 = 857 nM T59328 C3OBC6 134139548 IC50 = 61 nM T59328 C59COE 134139584 IC50 = 1.5 nM T59328 C81QJV 134139647 IC50 = 75 nM T59328 CW69GT 134139694 IC50 = 8 nM T59328 CQE08L 134139702 IC50 = 9 nM T59328 CK7EZ2 134139706 IC50 = 5.8 nM T59328 CO9W1Q 134139995 IC50 = 20 nM T59328 CHL7B1 134140023 IC50 > 1000 nM T59328 CJ9RI1 134140064 IC50 = 51 nM T59328 C8JR1X 134140108 IC50 = 7 nM T59328 C6M9DN 134140179 IC50 = 570 nM T59328 C1QSH4 134140222 IC50 = 1370 nM T59328 CCF0X1 134140501 IC50 = 0.65 nM T59328 C6UJG4 134140680 IC50 = 116 nM T59328 CI2L7Z 134140949 IC50 = 522 nM T59328 C1OB7Z 134141093 IC50 = 100.6 nM T59328 CFAW82 134141290 IC50 = 140 nM T59328 C6HD9W 134141630 IC50 = 53 nM T59328 CM05IQ 134141901 IC50 = 2 nM T59328 CLV6A3 134141947 IC50 = 24 nM T59328 C8KC5F 134142230 IC50 = 898 nM T59328 CS95WZ 134142314 IC50 = 9941 nM T59328 CP38FT 134142454 IC50 > 10000 nM T59328 CC3I0G 134142769 IC50 = 6400 nM T59328 CI92TY 134142809 IC50 = 870 nM T59328 C7TF6I 134142952 IC50 = 4.1 nM T59328 CJT12G 134143005 IC50 = 42 nM T59328 CY9M7L 134143068 IC50 = 747 nM T59328 CSTC29 134143257 IC50 = 509 nM T59328 C4F6VU 134143525 IC50 = 26 nM T59328 C92VFI 134143736 IC50 = 260 nM T59328 CZNJ57 134143863 IC50 = 4.6 nM T59328 CMV45A 134144196 IC50 = 2.7 nM T59328 CWS6V1 134144330 IC50 = 24 nM T59328 C0BJ1U 134144565 IC50 = 9.1 nM T59328 CGD4S5 134144603 IC50 = 28 nM T59328 CH1S3B 134144825 IC50 = 40.6 nM T59328 C38JMR 134145160 IC50 = 531 nM T59328 CO7LU3 134145579 IC50 = 383 nM T59328 CB89WK 134145650 IC50 > 10000 nM T59328 C0TYW7 134145741 IC50 = 388 nM T59328 C1OYR9 134145751 IC50 = 65 nM T59328 CBC06T 134145933 IC50 = 14 nM T59328 CVO98Y 134145943 IC50 > 100 nM T59328 CKZ2I0 134145988 IC50 = 593 nM T59328 CRZ0E5 134146010 IC50 = 8 nM T59328 CZP47U 134146163 IC50 = 160 nM T59328 CTMJ14 134146542 IC50 = 881 nM T59328 CN35SO 134146628 IC50 > 1000 nM T59328 CHJ13S 134146699 IC50 = 19 nM T59328 C0KNV3 134146887 IC50 = 3 nM T59328 CS7CJ4 134146891 IC50 = 212 nM T59328 C3K4ME 134147150 IC50 = 7 nM T59328 C4U8KT 134147234 IC50 = 7 nM T59328 CDF1R9 134147522 IC50 > 10000 nM T59328 CS0WH4 134147608 IC50 = 6.7 nM T59328 C5C9UN 134147625 IC50 = 140 nM T59328 CJ1FQ6 134147869 IC50 = 3 nM T59328 CXS38A 134147887 IC50 = 2 nM T59328 CUKE45 134147919 IC50 > 10000 nM T59328 C4ID3S 134148105 IC50 = 7 nM T59328 CZT40L 134148122 IC50 = 4 nM T59328 CZD10T 134148132 IC50 = 106 nM T59328 CPGL96 134148137 IC50 = 17 nM T59328 CDCJ80 134148182 IC50 > 1000 nM T59328 CN4HT6 134148374 IC50 = 330 nM T59328 CGVC01 134148454 IC50 = 714 nM T59328 CH8A5L 134148508 IC50 = 90 nM T59328 CH5O1F 134148524 IC50 = 15 nM T59328 C5R2PK 134148588 IC50 = 390 nM T59328 C0AWH3 134148660 IC50 = 10 nM T59328 CS0J8U 134148764 IC50 > 1000 nM T59328 CFZI08 134149229 IC50 = 817 nM T59328 C3AS1E 134149331 IC50 = 74 nM T59328 CP14DK 134149339 IC50 = 6.9 nM T59328 CRBI31 134149577 IC50 = 77 nM T59328 CIMW36 134149689 IC50 = 56 nM T59328 CU7FX1 134149906 IC50 = 6.3 nM T59328 C6B4YD 134149918 IC50 = 13 nM T59328 C6Z2JL 134149963 IC50 = 86 nM T59328 CE69LC 134150331 IC50 = 10 nM T59328 CIKN06 134150340 IC50 = 6.9 nM T59328 CQ03OC 134150381 IC50 = 10 nM T59328 CJ56EZ 134150417 IC50 = 1 nM T59328 CM7H0R 134150543 IC50 = 1.9 nM T59328 C1PDA8 134150559 IC50 = 470 nM T59328 CQK40B 134150618 IC50 = 10 nM T59328 C6CFO5 134150713 IC50 = 1 nM T59328 CA4SQ5 134151152 IC50 = 6 nM T59328 C76JIM 134151200 IC50 > 10000 nM T59328 C7CT2Y 134151327 IC50 = 61 nM T59328 CRH2V4 134151618 IC50 = 84 nM T59328 C7NB0Z 134152247 IC50 = 611 nM T59328 CU5T1N 134152381 IC50 > 10000 nM T59328 CG10PO 134152385 IC50 = 77 nM T59328 CI4A1T 134152401 IC50 = 12 nM T59328 CJ9N1A 134152440 IC50 = 14 nM T59328 C76WDH 134152470 IC50 = 44 nM T59328 CWT0Q7 134152512 IC50 > 100 nM T59328 CM62UF 134152586 IC50 = 103.4 nM T59328 C34KQM 134152648 IC50 = 6 nM T59328 C0N6JF 134152887 IC50 = 14 nM T59328 C9ORY0 134152991 IC50 = 21 nM T59328 CW6A7E 134153017 IC50 = 343 nM T59328 C5WV9Z 134153022 IC50 = 22 nM T59328 CLBK62 134153313 IC50 = 65 nM T59328 CLRD90 134153659 IC50 = 27 nM T59328 C1XJ7U 134153922 IC50 = 86 nM T59328 C6JFN5 134153988 IC50 = 72 nM T59328 CR09XE 134154074 IC50 = 88 nM T59328 C8Z3DN 134154342 IC50 = 21 nM T59328 C2Q1XW 134154347 IC50 = 36 nM T59328 CET5R1 134154580 IC50 = 184 nM T59328 C5YX7T 134154596 IC50 = 26 nM T59328 CTG04X 134154708 IC50 = 4 nM T59328 C07RWN 134154721 IC50 = 14 nM T59328 CV5M1T 134154754 IC50 = 5 nM T59328 CI0S4B 134155078 IC50 = 67 nM T59328 C2ISW7 134155088 IC50 = 1 nM T59328 CMH0X4 134155167 IC50 = 519 nM T59328 C48UIX 134155220 IC50 = 9 nM T59328 CVA34W 134155401 IC50 = 2 nM T59328 CR54HK 134155423 IC50 = 17 nM T59328 CJW2N9 134155488 IC50 = 1.1 nM T59328 C9DRQ6 134155700 IC50 = 60 nM T59328 C90IBM 134155874 IC50 = 9300 nM T59328 C6HN5J 134155932 IC50 = 12 nM T59328 CBY2R8 134156011 IC50 = 0.69 nM T59328 CS56YR 134156100 IC50 = 421 nM T59328 C4ZUO0 134156542 IC50 = 93 nM T59328 C2QN7B 134156570 IC50 = 2933 nM T59328 CKL8X3 134156658 IC50 = 45 nM T59328 CF7KA3 134156808 IC50 = 109 nM T59328 CQD93J 134156816 IC50 = 21 nM T59328 C3HCT6 134156845 IC50 = 25 nM T59328 CI4W7T 134156856 IC50 = 11.6 nM T59328 CH1GS2 134157091 IC50 = 6.5 nM T59328 COVM37 134157236 IC50 > 10000 nM T59328 CF85NI 134157315 IC50 = 205 nM T59328 CEHV70 134157345 IC50 = 19 nM T59328 CG36DX 134157614 IC50 = 127 nM T59328 C2AN7T 134611886 IC50 > 100000 nM T59328 CZ8W6R 134612705 IC50 > 1000 nM T59328 CYL5V1 134694986 IC50 > 30000 nM T59328 CG15PY 134812846 IC50 > 50000 nM T59328 CN3Y9J 134817166 IC50 = 1.1 nM T59328 COK96J 134827795 IC50 = 17 nM T59328 CIZ39M 134827836 IC50 > 100000 nM T59328 CJ04NP 134827837 IC50 = 140 nM T59328 C54FXD 134957362 IC50 > 10000 nM T59328 CUL3M1 134959408 Ki = 0.1 nM T59328 C82ENU 135128874 Ki = 105 nM T59328 C0NCM1 135236452 IC50 = 6.5 nM T59328 C7EMI6 135236457 IC50 = 210 nM T59328 CWBO79 135236483 IC50 = 219 nM T59328 CH3ZB7 135236498 IC50 = 5.8 nM T59328 CXDY80 135236566 IC50 = 9 nM T59328 C5SEK3 135236586 IC50 = 199 nM T59328 CIOD87 135236597 IC50 = 413 nM T59328 C45LFT 135236603 IC50 = 300 nM T59328 CR9TH8 135236627 IC50 > 10000 nM T59328 C3J5LM 135236635 IC50 = 20 nM T59328 CB6EG0 135236676 IC50 = 8630 nM T59328 CL93ZY 135236756 IC50 = 420 nM T59328 C0DV1Q 135236809 IC50 = 36 nM T59328 CS4BM3 135236903 IC50 = 10.9 nM T59328 CGJ07D 135236905 IC50 = 48 nM T59328 CNC56O 135251923 IC50 = 26.8 nM T59328 C2PH4R 135251924 IC50 = 494 nM T59328 CO43PJ 135251926 IC50 = 730 nM T59328 C4IO8Z 135313938 Ki = 0.03 nM T59328 C6IYG1 135314117 IC50 < 1 nM T59328 CCM74D 135369110 IC50 = 46.5 nM T59328 C4PN7O 135400972 IC50 = 50000 nM T59328 CVJK60 135402835 IC50 = 6 nM T59328 CPE8O5 135402837 IC50 = 588 nM T59328 CO3H4I 135402838 IC50 = 0.17 nM T59328 CK67RJ 135402839 IC50 = 4.7 nM T59328 C05WPI 135402840 IC50 = 1.24 nM T59328 C38ASJ 135402848 IC50 = 346.74 nM T59328 CLFE42 135402849 IC50 = 1.6 nM T59328 CJ1I5M 135402981 IC50 > 1000 nM T59328 CH97JB 135402982 IC50 > 1000 nM T59328 C26GSU 135402983 IC50 > 1000 nM T59328 CK8EJ6 135402984 IC50 > 1000 nM T59328 C1Q9SE 135407125 IC50 = 130000 nM T59328 CAZ5X6 135407149 IC50 = 60000 nM T59328 CR3XN0 135408977 IC50 = 3100 nM T59328 C7LI1N 135408978 IC50 = 1400 nM T59328 CQ54JK 135410197 IC50 = 71700 nM T59328 CQ4RD2 135410274 IC50 > 10000 nM T59328 CUI1B3 135417010 IC50 = 7700 nM T59328 CK9D4A 135428921 EC50 = 33000 nM T59328 C85SLV 135430346 IC50 = 20 ug.mL-1 T59328 COI9Y2 135431544 IC50 = 5300 nM T59328 CU60YC 135431661 IC50 > 30000 nM T59328 C5FO9E 135433976 IC50 = 30000 nM T59328 C4VH8I 135438239 IC50 = 5600 nM T59328 C16XLU 135454992 IC50 > 10000 nM T59328 CIP6W1 135457450 IC50 = 10000 nM T59328 CIJ9Q2 135461535 IC50 = 3920 nM T59328 C3WK8O 135464283 IC50 = 61000 nM T59328 CX35PB 135468746 IC50 > 100000 nM T59328 C01NXG 135469322 IC50 = 58000 nM T59328 CMU4G6 135474309 IC50 = 27000 nM T59328 CWPK94 135478626 IC50 = 1400 nM T59328 CRTS92 135484881 IC50 > 100000 nM T59328 CGXS54 135485502 IC50 = 75000 nM T59328 CMOR61 135492395 IC50 > 10000 nM T59328 CKF6R5 135492549 IC50 >> 2000 nM T59328 CJB83H 135494293 IC50 = 6 ug.mL-1 T59328 CCOL98 135499946 IC50 = 100000 nM T59328 C64EMD 135500075 IC50 > 10000 nM T59328 CH91IT 135503554 IC50 > 10000 nM T59328 CP0R1O 135503606 IC50 > 100000 nM T59328 CVZ08D 135509841 IC50 > 10000 nM T59328 CYQ5M6 135511836 IC50 = 300000 nM T59328 CGI1H3 135516745 IC50 = 20000 nM T59328 C5TW9S 135517293 IC50 >> 10000 nM T59328 CG1WR0 135518082 IC50 = 130000 nM T59328 CJI0G1 135520135 IC50 > 10000 nM T59328 CLK9D1 135523696 IC50 = 75000 nM T59328 CTJ48K 135524085 IC50 = 3300 nM T59328 CUT1W7 135524168 IC50 > 10000 nM T59328 CRT3X6 135524445 IC50 = 2100 nM T59328 CIA18F 135525349 IC50 = 5000 nM T59328 CIM0Q6 135526986 IC50 > 20000 nM T59328 C3XK7R 135531249 IC50 = 8.5 ug.mL-1 T59328 C2MAC7 135536640 IC50 > 100000 nM T59328 COXH29 135543616 IC50 >> 20000 nM T59328 CM72XH 135546247 IC50 = 20 ug.mL-1 T59328 C0J3BN 135678111 IC50 > 50000 nM T59328 CU29YK 135750268 IC50 = 922 nM T59328 CX4ZB3 135863110 IC50 > 10000 nM T59328 CM3UC9 135883136 IC50 = 370 nM T59328 C8LN7E 135883350 IC50 > 100000 nM T59328 CUV73C 135883354 IC50 > 100000 nM T59328 CIPA79 135937899 IC50 = 2200 nM T59328 C12UDA 135947972 IC50 = 1040 nM T59328 CN42ZS 135947973 IC50 = 954 nM T59328 CF8AO3 135947974 IC50 = 6900 nM T59328 CW08GJ 135947976 IC50 = 7400 nM T59328 CJN7E2 135947978 IC50 = 908 nM T59328 CFKH34 135947979 IC50 = 88 nM T59328 C2PAV1 135971426 IC50 = 3300 nM T59328 C9W6BT 136002660 IC50 = 10900 nM T59328 CD9CT6 136002661 IC50 = 989 nM T59328 C4T9KZ 136002662 IC50 = 726 nM T59328 CHA4N2 136013680 IC50 > 10 nM T59328 CLN6Y8 136026516 IC50 > 100000 nM T59328 CQ0KD1 136036218 IC50 = 1.585 nM T59328 CGP0K5 136036219 IC50 = 0.4169 nM T59328 C2ZX7P 136036220 IC50 = 0.912 nM T59328 C4HNF6 136036221 IC50 = 5.754 nM T59328 C67UGS 136036222 IC50 = 3.631 nM T59328 CLZ9Q1 136036223 IC50 = 0.4786 nM T59328 C3N4KU 136036228 IC50 = 0.7244 nM T59328 C5AY0R 136036229 IC50 = 0.7762 nM T59328 CH0AO1 136042228 IC50 = 34250 nM T59328 CJ7U4C 136053657 IC50 > 100000 nM T59328 CZP3W5 136066077 IC50 = 28.5 nM T59328 C8D0YV 136066078 IC50 = 3.16 nM T59328 C4LGS1 136066079 IC50 = 65.5 nM T59328 CCAM43 136066080 IC50 = 4.45 nM T59328 CIG6B4 136066100 IC50 = 16.9 nM T59328 CBH08O 136066101 IC50 = 23.8 nM T59328 CG1R7B 136087060 IC50 > 10000 nM T59328 CGP69Y 136130281 IC50 = 501187.23 nM T59328 CH64ID 136175114 IC50 > 10000 nM T59328 CDT7E4 136211077 IC50 > 1000 nM T59328 C9RE8D 136215817 IC50 > 100000 nM T59328 C1YUD0 136219394 IC50 > 10 nM T59328 C5QAT2 136236302 IC50 = 24.1 nM T59328 CIU8W3 136254389 IC50 > 10 nM T59328 CRK8E5 136391507 IC50 = 0.48 nM T59328 CR69AU 136928128 IC50 = 0.63 nM T59328 C03VDE 136928142 IC50 = 141 nM T59328 CTAS87 136983688 IC50 = 2.1 nM T59328 C8M2DL 136983691 IC50 = 169 nM T59328 CMOH82 136983718 IC50 = 0.18 nM T59328 C1JSX0 136983721 IC50 = 0.46 nM T59328 CRE05Z 136983730 IC50 = 3.1 nM T59328 CMP62O 136983732 IC50 = 0.3 nM T59328 CB26DO 136983736 IC50 = 0.66 nM T59328 C9J5KZ 136983740 IC50 = 0.34 nM T59328 CN7W2C 136983741 IC50 = 1.2 nM T59328 CPM64E 136983746 IC50 = 0.79 nM T59328 CM2IO7 136983748 IC50 < 0.25 nM T59328 C60HNV 136983761 IC50 = 3.2 nM T59328 C4EKW0 136983767 IC50 = 21 nM T59328 C69LHV 137175062 Ki = 58 nM T59328 C41AYR 137175217 Ki = 88 nM T59328 C83WAK 137189946 IC50 = 3600 nM T59328 C0LR2H 137189948 IC50 > 20000 nM T59328 C8KW0I 137189951 IC50 = 3450 nM T59328 COX23B 137189952 IC50 = 4390 nM T59328 CSGM03 137210056 IC50 > 10000 nM T59328 CXT8B9 137287443 IC50 = 51 nM T59328 C2SY8T 137302575 IC50 = 3 nM T59328 CUL6Z7 137319850 IC50 < 1 nM T59328 C3Z4AT 137321159 IC50 > 10000 nM T59328 CE75QD 137321162 IC50 = 520 nM T59328 CM4TU2 137321167 IC50 = 30 nM T59328 CWH6I2 137348469 IC50 = 2.5 nM T59328 CF2B4A 137348470 IC50 = 1 nM T59328 CKC2Q5 137348686 IC50 = 649 nM T59328 C6A8BE 137349495 IC50 = 690 nM T59328 C9OQ2L 137436777 IC50 = 168.8 nM T59328 CPYC42 137436898 IC50 > 1000 nM T59328 CZL7X1 137436936 IC50 = 65.1 nM T59328 C1KSZ6 137475463 IC50 = 5882 nM T59328 C2FT1L 137475480 IC50 = 6863 nM T59328 C13DTZ 137628688 IC50 = 5.8 nM T59328 C6V3UK 137631426 IC50 = 11.3 nM T59328 C58XRH 137631553 IC50 = 23.99 nM T59328 CZE86J 137631564 IC50 = 183 nM T59328 CMP5H4 137631852 IC50 > 10000 nM T59328 C0CE4R 137631936 IC50 = 2 nM T59328 C81MHK 137631947 IC50 = 48.9 nM T59328 C25ERN 137631967 IC50 = 4.2 nM T59328 CK9TO3 137632059 IC50 = 10.2 nM T59328 CH9WK1 137632228 IC50 > 10000 nM T59328 CW2I0X 137632429 IC50 = 28.9 nM T59328 C6HYQ4 137632485 IC50 = 373.7 nM T59328 CNO0W6 137632514 IC50 = 46 nM T59328 C6BWP9 137632530 IC50 = 297 nM T59328 C8YXN5 137632579 IC50 = 10.2 nM T59328 C9Y4UW 137632652 IC50 = 15.4 nM T59328 CX4BG3 137632686 IC50 = 257 nM T59328 C1IRD9 137632976 IC50 = 600 nM T59328 COW53U 137633148 IC50 = 60.1 nM T59328 C8J5YE 137633149 IC50 = 60953.69 nM T59328 C52PDU 137633245 IC50 = 100000 nM T59328 CAW72M 137633292 IC50 = 3400 nM T59328 CWP23Z 137633367 IC50 = 5700 nM T59328 C6W9VB 137633473 IC50 < 1 nM T59328 CKD94A 137633488 IC50 = 65400 nM T59328 CFUY16 137633842 IC50 = 4300 nM T59328 C41TLP 137634049 IC50 = 188.2 nM T59328 CNX0F9 137634126 IC50 = 360 nM T59328 CHC70D 137634143 IC50 = 725.3 nM T59328 C3Z5UO 137634208 IC50 = 8470 nM T59328 CI1E8V 137634241 IC50 > 10000 nM T59328 CE9G6I 137634299 IC50 = 120 nM T59328 CD64EL 137634342 IC50 = 25.3 nM T59328 C58JAF 137634409 IC50 = 549.6 nM T59328 CFP2A7 137634412 IC50 = 100000 nM T59328 CM3JB8 137634462 IC50 > 150 nM T59328 CP0J4V 137634715 IC50 = 10 nM T59328 C42PMG 137634834 IC50 = 52.8 nM T59328 C2DT0F 137634837 IC50 = 413 nM T59328 C9MJB3 137635188 IC50 = 17.6 nM T59328 CKH35C 137635255 Ki = 3680 nM T59328 C18FSE 137635348 IC50 = 28.7 nM T59328 CICR67 137635590 IC50 = 14.2 nM T59328 C42CPG 137635606 IC50 < 1 nM T59328 CS23KQ 137635618 IC50 = 20000 nM T59328 CY4M7O 137635632 Ki = 640 nM T59328 CI8T3V 137635635 IC50 = 1120 nM T59328 C5JD9N 137635898 IC50 = 2.3 nM T59328 C61KRW 137636025 IC50 = 5900 nM T59328 CW03UM 137636140 IC50 = 10 nM T59328 C1UM2S 137636157 IC50 > 150 nM T59328 CL4US7 137636248 IC50 > 150 nM T59328 C6LB3K 137636403 IC50 = 100000 nM T59328 CY6S7J 137636429 IC50 = 26.9 nM T59328 CVD9E7 137636479 IC50 = 60 nM T59328 C1EXD3 137636509 IC50 = 67.9 nM T59328 CB89IY 137636527 IC50 > 100000 nM T59328 CPF75D 137636602 IC50 = 55.5 nM T59328 C2IOU5 137636607 IC50 = 26 nM T59328 CXLM63 137636621 IC50 < 0.3 nM T59328 C2FA3S 137636658 IC50 = 4050 nM T59328 CT17QN 137636787 IC50 = 2.3 nM T59328 C8BDC7 137636863 IC50 = 7 nM T59328 C9K5AS 137637051 IC50 = 28 nM T59328 C06JRX 137637094 IC50 = 4.7 nM T59328 CXJ3Q0 137637114 IC50 = 6.13 nM T59328 CRD5K6 137637150 IC50 = 20 nM T59328 CB9MO6 137637177 IC50 = 1.8 nM T59328 C5LU2S 137637274 Ki = 80 nM T59328 CSC2Q3 137637327 IC50 = 12 nM T59328 C0YD2I 137637558 IC50 = 467 nM T59328 CJ86NK 137637579 IC50 = 55 nM T59328 C63SHA 137637655 IC50 = 56 nM T59328 CT7BW5 137637707 IC50 < 1 nM T59328 C36UDX 137637748 IC50 = 25 nM T59328 CRXH80 137637913 IC50 = 1 nM T59328 CIPT52 137638089 IC50 = 0.5 nM T59328 CGNL27 137638186 IC50 = 1.9 nM T59328 CSU32D 137638440 IC50 = 7.8 nM T59328 CD7ZQ9 137638445 IC50 = 120 nM T59328 CU24QC 137638448 IC50 = 33.6 nM T59328 C4NBP2 137638482 IC50 = 11.2 nM T59328 CI45NR 137638579 IC50 = 133.1 nM T59328 CDHR26 137638664 IC50 = 1300 nM T59328 CSC8I9 137638715 IC50 = 120 nM T59328 CG09DY 137638779 IC50 = 27.4 nM T59328 CIAL90 137638797 IC50 < 1 nM T59328 C8G0XY 137638840 IC50 = 97 nM T59328 C3FU9S 137638860 IC50 = 436.3 nM T59328 CS8I4L 137639015 IC50 = 595.2 nM T59328 CB9K0T 137639063 IC50 > 150 nM T59328 CLWZ62 137639100 IC50 = 1.6 nM T59328 CLM2E7 137639118 IC50 < 0.3 nM T59328 CDG3W9 137639160 Ki = 5950 nM T59328 C1CJL8 137639161 IC50 = 302 nM T59328 CTQ2Y9 137639273 IC50 > 150 nM T59328 CM12TX 137639299 IC50 = 36.8 nM T59328 CZ4JS5 137639379 Ki = 370 nM T59328 CE75PY 137639383 IC50 = 3.3 nM T59328 CBM75H 137639408 IC50 = 35.8 nM T59328 C39GHY 137639513 Ki = 0.38 nM T59328 C3UBE2 137639638 IC50 = 47.1 nM T59328 CE96AL 137639657 IC50 = 3.2 nM T59328 CEWX78 137639774 IC50 = 34320 nM T59328 C9QS8P 137639893 IC50 > 150 nM T59328 C0GI7M 137639998 Ki = 290 nM T59328 CZ3RG6 137640107 IC50 = 28.3 nM T59328 CUQ32R 137640370 IC50 = 1.9 nM T59328 CP4WE6 137640788 IC50 = 4.53 nM T59328 CEPC29 137640799 IC50 = 220 nM T59328 C3PBM5 137640804 IC50 = 20 nM T59328 CZA04C 137640806 IC50 = 2000 nM T59328 C6LE5P 137640904 Ki = 610 nM T59328 C45TDX 137641093 IC50 = 287 nM T59328 CI9A6R 137641259 IC50 = 26.5 nM T59328 CF0B2T 137641286 IC50 = 137 nM T59328 C7TG3J 137641313 IC50 > 19952.62 nM T59328 CM0ID8 137641315 IC50 = 100000 nM T59328 C2S5HW 137641579 IC50 = 200 nM T59328 CADV57 137641678 IC50 = 22 nM T59328 CC7NA3 137641695 IC50 = 7.6 nM T59328 C4S0NY 137641776 IC50 = 20 nM T59328 CDF05B 137641797 IC50 = 1600 nM T59328 CI48MT 137641870 IC50 = 15.69 nM T59328 CO7T1M 137642099 IC50 = 35.4 nM T59328 CA26QR 137642204 IC50 = 217 nM T59328 CE78MV 137642234 IC50 = 10 nM T59328 CFP6S7 137642384 IC50 = 132.1 nM T59328 C0M2DV 137642413 IC50 = 2900 nM T59328 CHSF21 137642481 IC50 = 6 nM T59328 CYIM43 137642492 IC50 = 46300 nM T59328 CG0P7F 137642583 IC50 < 0.3 nM T59328 C1BEM9 137642718 IC50 = 0.8 nM T59328 CR7DU4 137642765 Ki = 910 nM T59328 C04WMX 137642837 IC50 < 1 nM T59328 C86ZQY 137642882 IC50 = 46.8 nM T59328 CU6V4B 137642950 IC50 = 86200 nM T59328 CU8YX6 137643005 IC50 = 167300 nM T59328 CEX71A 137643024 IC50 = 889 nM T59328 C3VE1J 137643259 IC50 = 19.3 nM T59328 CC24DF 137643392 IC50 = 838.5 nM T59328 C1TN5U 137643437 IC50 = 127.8 nM T59328 CO2WA8 137643441 IC50 = 1.1 nM T59328 C5NB8J 137643535 IC50 = 100000 nM T59328 CSJ4F0 137643599 IC50 = 295.7 nM T59328 C9KC1X 137643767 IC50 = 2626 nM T59328 CZN72T 137644087 IC50 = 222.5 nM T59328 CRQL24 137644097 IC50 = 100000 nM T59328 CNK3C1 137644195 IC50 = 24.4 nM T59328 CGV72K 137644347 IC50 > 150 nM T59328 CV8G5N 137644357 IC50 < 1 nM T59328 CJ6I3O 137644466 IC50 = 1.1 nM T59328 CVP54C 137644489 IC50 = 6.2 nM T59328 CQ08RW 137644617 IC50 = 365 nM T59328 CMEL14 137644727 Ki = 270 nM T59328 CD29JK 137644944 IC50 = 145 nM T59328 C0CSA2 137645004 IC50 = 4.9 nM T59328 COQ1G5 137645019 IC50 = 1.79 nM T59328 CMA01W 137645075 IC50 = 22.2 nM T59328 CS03JL 137645107 IC50 = 60 nM T59328 C15SPX 137645121 IC50 = 100000 nM T59328 CZDI94 137645280 IC50 = 1900 nM T59328 CCG29K 137645358 IC50 = 3210 nM T59328 CKP7N9 137645385 Ki = 1260 nM T59328 C27ISW 137645443 IC50 = 60.7 nM T59328 C37UPA 137645513 IC50 = 40 nM T59328 C9RY1I 137645557 IC50 = 16 nM T59328 CW5N0Q 137645598 IC50 = 40 nM T59328 C7Q0KP 137645669 IC50 = 373 nM T59328 CJ94TQ 137645832 IC50 = 7230 nM T59328 CQJ45H 137645835 IC50 = 26.6 nM T59328 CT4JK0 137645956 IC50 = 14.5 nM T59328 C03VKP 137646019 IC50 < 1 nM T59328 CFVP34 137646278 Ki = 110 nM T59328 CHL6W7 137646293 IC50 = 36.9 nM T59328 CX9QM0 137646296 Ki = 900 nM T59328 CN2J6Z 137646310 IC50 = 365 nM T59328 C7K6XE 137646529 IC50 > 10000 nM T59328 CDK1X9 137646546 IC50 = 3400 nM T59328 CSEV89 137646548 IC50 = 45 nM T59328 CS6J0V 137646549 IC50 = 98 nM T59328 CB45FK 137646625 IC50 = 15 nM T59328 C1MJ2B 137646681 IC50 = 2.6 nM T59328 C39ECO 137646754 IC50 = 33189.45 nM T59328 CE2GS1 137646967 IC50 = 117.5 nM T59328 CNR6Y9 137647154 IC50 = 427.7 nM T59328 C84XPS 137647374 IC50 = 63.6 nM T59328 CRI7W4 137647547 IC50 = 25.5 nM T59328 C1MO6F 137647858 IC50 = 153 nM T59328 CV34AT 137647876 IC50 = 4700 nM T59328 CB4G7L 137648004 IC50 = 979.49 nM T59328 CHKS97 137648071 Ki = 90 nM T59328 CB02WE 137648106 IC50 = 87 nM T59328 CHYD27 137648384 IC50 = 10.9 nM T59328 C4Q5FE 137648385 IC50 < 0.5 nM T59328 CZO42N 137648629 IC50 > 100000 nM T59328 CDWM98 137648631 IC50 = 209 nM T59328 CNZV16 137648828 IC50 = 4.5 nM T59328 CA1H0Y 137649110 IC50 = 18.7 nM T59328 CPY41L 137649188 IC50 = 102 nM T59328 CQ53DI 137649227 IC50 = 210 nM T59328 CQ2D4K 137649247 IC50 = 8.9 nM T59328 CRL38H 137649329 IC50 = 146.3 nM T59328 CWAP61 137649410 IC50 = 24 nM T59328 CZ5DB2 137649455 IC50 = 9.5 nM T59328 C3XQ4T 137649572 IC50 = 20 nM T59328 C68MVW 137649573 IC50 = 148 nM T59328 CTBG10 137649803 IC50 = 208.4 nM T59328 CG3D9R 137649880 IC50 = 6.7 nM T59328 CR5JN8 137649915 IC50 = 462 nM T59328 CN3I0J 137650029 IC50 = 130 nM T59328 C6JIK5 137650097 IC50 < 1 nM T59328 CZ5VL9 137650197 IC50 = 100000 nM T59328 CH2R1F 137650251 IC50 = 780 nM T59328 C3UBN8 137650330 IC50 = 3700 nM T59328 CR27SL 137650383 IC50 = 39700 nM T59328 CQ4R1I 137650454 IC50 = 286 nM T59328 CI1U0H 137650532 IC50 = 9.2 nM T59328 C1A6ZV 137650580 IC50 = 218 nM T59328 CX12DJ 137650597 IC50 = 7.2 nM T59328 C4N2VA 137650617 IC50 = 144 nM T59328 C12JHN 137650629 IC50 = 12.1 nM T59328 CS0D7H 137650797 IC50 = 97 nM T59328 CV7WE6 137651016 IC50 = 258 nM T59328 CO6DY4 137651084 IC50 = 2500 nM T59328 C9CZ5R 137651233 IC50 = 22 nM T59328 CM2WA6 137651258 IC50 = 421 nM T59328 C5ZEI9 137651283 IC50 > 150 nM T59328 CX9BD8 137651363 IC50 = 3100 nM T59328 C1DK0P 137651391 IC50 = 8.1 nM T59328 C0IY3L 137651740 IC50 < 1 nM T59328 CUN78O 137651765 IC50 = 5 nM T59328 CBP7D8 137651768 IC50 = 1300 nM T59328 CR0QK4 137651864 IC50 = 15.8 nM T59328 C0GB7L 137651865 IC50 = 1300 nM T59328 CU1WH2 137651878 IC50 = 5.6 nM T59328 C3X0VR 137652014 IC50 = 73500 nM T59328 C2QMD3 137652087 IC50 = 55 nM T59328 C28VPE 137652194 IC50 = 10.71 nM T59328 C6PQ3M 137652198 IC50 = 12 nM T59328 CQUY83 137652218 IC50 = 8300 nM T59328 CO41DK 137652335 IC50 = 673 nM T59328 C7SB9W 137652377 IC50 = 20.6 nM T59328 CJ6S9T 137652622 IC50 = 8.5 nM T59328 C1E0GD 137652646 IC50 = 8.1 nM T59328 CX2L6R 137652830 IC50 = 13 nM T59328 C7Z3OK 137652842 IC50 = 2400 nM T59328 CIK69O 137652848 IC50 = 1.6 nM T59328 CDJ1E5 137652860 IC50 = 1100 nM T59328 C28QUP 137652864 IC50 = 642.7 nM T59328 CW39CF 137652891 IC50 = 57 nM T59328 C3LAD6 137652990 IC50 = 1021 nM T59328 CNB10S 137653041 IC50 = 4900 nM T59328 C9BF1E 137653143 IC50 = 25000 nM T59328 C6RWG4 137653308 IC50 = 4500 nM T59328 CMS31R 137653327 IC50 = 32.35 nM T59328 CZLB29 137653418 IC50 = 100000 nM T59328 C5LV3R 137653430 IC50 = 11 nM T59328 CVF8B2 137653486 IC50 = 9.1 nM T59328 CWFI42 137653795 IC50 = 69984.2 nM T59328 CX3JS6 137653952 IC50 = 278.2 nM T59328 CRSC07 137654213 IC50 = 55.5 nM T59328 CDIG10 137654476 IC50 = 91.8 nM T59328 CHL6R9 137654533 IC50 < 1 nM T59328 C7UEM1 137654543 IC50 = 50000 nM T59328 CUP85I 137654607 IC50 = 518 nM T59328 CST9Z6 137654612 IC50 = 1.2 nM T59328 CZ1D3X 137654743 IC50 > 150 nM T59328 CPMI90 137654861 IC50 = 11 nM T59328 C5CH2P 137654954 IC50 = 216.1 nM T59328 CQGX68 137655106 IC50 = 11.4 nM T59328 CHR5Y4 137655134 IC50 = 29.4 nM T59328 CRN09J 137655337 IC50 = 76 nM T59328 CCXH57 137655416 Ki = 640 nM T59328 C9JT1N 137655519 IC50 = 20800 nM T59328 CO03SP 137655672 IC50 = 32.1 nM T59328 CJHR85 137655678 IC50 = 6900 nM T59328 C5OEN8 137655763 IC50 > 150 nM T59328 CF4BR6 137655863 IC50 = 715 nM T59328 C56LGP 137655890 IC50 = 83.82 nM T59328 CP0EK1 137656130 IC50 > 150 nM T59328 CJ1AL4 137656216 IC50 = 362 nM T59328 C4OL7J 137656236 Ki = 4030 nM T59328 CF65SR 137656304 IC50 = 112.4 nM T59328 CBUK30 137656424 IC50 = 45081.67 nM T59328 CM1X2Z 137656744 IC50 = 5000 nM T59328 COZA85 137656751 IC50 = 80.91 nM T59328 CIP0S1 137656884 IC50 = 10 nM T59328 C02CKX 137656919 IC50 = 888.2 nM T59328 CGK74V 137657167 IC50 = 4.87 nM T59328 CEX13S 137657186 IC50 = 8.9 nM T59328 CKVO51 137657233 IC50 = 4.9 nM T59328 CE2F4M 137657262 IC50 = 383 nM T59328 C4U6BC 137657356 IC50 = 2500 nM T59328 C4L3EC 137657481 IC50 = 0.07 nM T59328 CE3KR1 137657520 IC50 > 150 nM T59328 CWE31H 137657545 IC50 = 417 nM T59328 C2W5XI 137657580 IC50 = 24.9 nM T59328 CV5H3Z 137657932 IC50 = 3.1 nM T59328 CZP9J1 137658032 IC50 = 224.5 nM T59328 C2MCK3 137658120 IC50 = 22 nM T59328 CS14VU 137658122 IC50 = 1200 nM T59328 C64HKO 137658202 IC50 = 23700 nM T59328 CGP0F8 137658204 IC50 < 1 nM T59328 CNM0R5 137658207 IC50 = 0.6 nM T59328 CPV1S9 137658287 IC50 > 1000 nM T59328 CCOQ25 137658337 IC50 = 6.8 nM T59328 CW59EN 137658341 IC50 = 27 nM T59328 C1W3SU 137658355 IC50 = 6.8 nM T59328 CO41NV 137658479 IC50 > 100000 nM T59328 C0T6DR 137658736 IC50 = 19.5 nM T59328 C7IVT9 137658762 IC50 = 167.1 nM T59328 CW89GI 137658864 IC50 < 1 nM T59328 CPD68B 137658974 IC50 > 150 nM T59328 CH5JU3 137658981 IC50 = 23.6 nM T59328 CV2L4Q 137659016 IC50 < 1 nM T59328 C7PL9R 137659061 IC50 = 55.5 nM T59328 CR91LE 137659218 IC50 = 5.7 nM T59328 C2GN1V 137659253 IC50 = 80 nM T59328 C0DC5L 137659278 Ki = 520 nM T59328 CE93JS 137659304 IC50 = 10 nM T59328 CJF6G7 137659313 IC50 = 1100 nM T59328 CC54PL 137659460 IC50 = 17.7 nM T59328 CS61AX 137659496 Ki = 5670 nM T59328 C4HZM7 137659498 IC50 > 150 nM T59328 CJ4YM8 137659634 IC50 = 3.4 nM T59328 C8NZ9V 137659669 IC50 = 75 nM T59328 C73CXG 137659722 IC50 = 15.7 nM T59328 CKL97P 137659725 IC50 = 23.4 nM T59328 CT94YA 137659769 IC50 = 32.1 nM T59328 CS43UI 137659891 IC50 = 15.8 nM T59328 CX2PB5 137660250 IC50 > 150 nM T59328 CBTU32 137660306 IC50 = 360 nM T59328 C46WON 137660327 IC50 > 1000 nM T59328 CLIB19 137660335 IC50 = 33.2 nM T59328 C07JTH 137660356 Ki = 1870 nM T59328 CF41AQ 137660592 IC50 = 4.9 nM T59328 CR4N5S 137660661 IC50 = 1.5 nM T59328 CTZ05I 137660747 IC50 = 11.42 nM T59328 C98GQX 137660836 IC50 = 8.7 nM T59328 C0YZP2 137660958 IC50 < 1 nM T59328 CCO5E1 137660978 IC50 = 10 nM T59328 C89EDU 137661037 IC50 = 6100 nM T59328 C9T8DS 137661049 IC50 = 22 nM T59328 CJ52DB 137661068 IC50 < 1 nM T59328 C1L7BC 137661158 IC50 = 1.9 nM T59328 CKY35O 137661181 Ki = 120 nM T59328 C7PQ6B 137661273 IC50 > 150 nM T59328 CMSH35 137661302 IC50 = 216 nM T59328 CSOE96 137661336 IC50 = 71.6 nM T59328 CM0N3T 137661420 IC50 = 2.6 nM T59328 C2EJB9 137661577 IC50 = 377 nM T59328 CYVS73 137661698 IC50 = 13 nM T59328 CB72MA 137661754 IC50 = 45000 nM T59328 C25FCZ 137661759 IC50 = 33 nM T59328 CT43IF 137661858 IC50 = 1.1 nM T59328 C0Y4XD 137662183 IC50 = 3900 nM T59328 CUY09E 137662185 IC50 = 626 nM T59328 C6CZA9 137662310 IC50 = 700 nM T59328 CM3UF7 137700779 IC50 > 10000 nM T59328 CT1D9K 138454747 IC50 > 1000000 nM T59328 C5LQU9 138479230 IC50 = 384.8 nM T59328 CSRI06 138547901 IC50 > 1000 nM T59328 CUXO19 138617501 IC50 > 1000 nM T59328 C9NYR2 138911325 IC50 = 27.5 nM T59328 CRWA29 139030520 IC50 > 2000 nM T59328 CJI5X1 139447554 IC50 = 12 nM T59328 CDQS68 139447649 IC50 = 519 nM T59328 CSDG73 139447864 IC50 = 353 nM T59328 CZ85HW 139593668 IC50 = 2100 nM T59328 CNI84L 139593669 IC50 = 267 nM T59328 COB9P2 141456067 IC50 > 10000 nM T59328 CWKN18 141489617 IC50 = 7.7 nM T59328 CZ6OQ4 141489621 IC50 = 33.1 nM T59328 C2V3CZ 141489622 IC50 = 142.7 nM T59328 CA6ZE3 141489625 IC50 = 202.3 nM T59328 CTG0M3 141489626 IC50 = 838.5 nM T59328 C42QLX 141489627 IC50 = 38.5 nM T59328 CH74WV 141489632 IC50 > 1000 nM T59328 C8YS7B 141489636 IC50 = 4.1 nM T59328 CZB56Q 141489640 IC50 = 4.1 nM T59328 C9X3BQ 141494014 IC50 = 53.2 nM T59328 CUG0M7 141494019 IC50 = 9.9 nM T59328 CUFX86 141494026 IC50 = 1.5 nM T59328 C4YTS8 141494027 IC50 = 12 nM T59328 CP6ZN9 141494035 IC50 = 1.6 nM T59328 C27MYX 141494043 IC50 = 85 nM T59328 CMND29 141494046 IC50 = 3.9 nM T59328 CT1EH2 141494048 IC50 = 6.5 nM T59328 CHO81S 141494057 IC50 = 3.3 nM T59328 C3SI7W 141494065 IC50 = 2.7 nM T59328 CEVI18 141494066 IC50 = 28.8 nM T59328 CP19EN 141509386 IC50 = 4 nM T59328 CCXT19 141510925 IC50 = 892 nM T59328 C9ED8K 141510928 IC50 = 556 nM T59328 C7TW9O 141510929 IC50 = 114 nM T59328 COLJ50 141510933 IC50 = 104 nM T59328 CI5KY6 141510937 IC50 = 805 nM T59328 CP20DC 141515864 IC50 = 7 nM T59328 CU17OE 141515867 IC50 = 20.7 nM T59328 C34CKN 141523354 IC50 > 10000 nM T59328 CTR7D4 141535114 IC50 = 42.3 nM T59328 CF1R6Z 141725864 IC50 = 7.8 nM T59328 CK35HM 141726486 IC50 = 3.62 nM T59328 C1QB4I 141740774 IC50 = 985 nM T59328 C9T0WU 141740777 IC50 = 37 nM T59328 C4DY2A 141740778 IC50 = 7.5 nM T59328 CMA73H 141740779 IC50 = 1621 nM T59328 COSZ17 141740780 IC50 = 201 nM T59328 CFV8J1 141740781 IC50 = 892 nM T59328 CKIY74 141740782 IC50 > 2000 nM T59328 CEWT18 141740783 IC50 = 977 nM T59328 C7PGK2 141740785 IC50 = 923 nM T59328 CF9N8G 141740786 IC50 = 684 nM T59328 C9XKQ7 141740787 IC50 > 2000 nM T59328 C7M4FY 141740788 IC50 = 1689 nM T59328 C67AUS 141740789 IC50 = 360 nM T59328 CNA8J2 141740790 IC50 = 1128 nM T59328 C72PLS 141740792 IC50 = 16 nM T59328 CYU95H 141740794 IC50 = 203 nM T59328 C1Y4TJ 141740795 IC50 = 998 nM T59328 C62QXI 141740796 IC50 = 20 nM T59328 CDEX12 142518169 IC50 = 81.7 nM T59328 CCXG67 142735680 IC50 = 6 nM T59328 CP17MF 142747584 IC50 = 23 nM T59328 CGRY21 142747612 IC50 = 46 nM T59328 CQ15DI 142747615 IC50 = 38.7 nM T59328 C9THY0 145314346 IC50 = 257 nM T59328 CMHX97 145331319 IC50 = 1.4 nM T59328 CVID46 145331320 IC50 = 68 nM T59328 CW1P9K 145331325 IC50 = 81 nM T59328 CDB9Y1 145331327 IC50 = 2.5 nM T59328 CG6V5Q 145331334 IC50 = 17 nM T59328 CGPH07 145331338 IC50 = 4.7 nM T59328 C6C5DF 145331339 IC50 = 0.6 nM T59328 CXCO76 145331341 IC50 = 1.3 nM T59328 CO9P7G 145351804 IC50 > 1000 nM T59328 C6VB3O 145925651 IC50 >= 5000 nM T59328 C29XUO 145945978 IC50 > 1000 nM T59328 C91UGF 145946092 IC50 = 39 nM T59328 C4HB8M 145949394 IC50 = 812 nM T59328 CB3Z1W 145949428 IC50 = 8.7 nM T59328 CTR3F0 145949484 IC50 = 4 nM T59328 CK4N8D 145951329 IC50 = 71 nM T59328 C9TJ8F 145951621 IC50 = 174.5 nM T59328 CH8K2T 145952204 IC50 = 4100 nM T59328 CM3CX8 145952650 IC50 = 890 nM T59328 CKRP30 145952676 IC50 = 110 nM T59328 C8V4MP 145952681 IC50 = 865 nM T59328 CNI31W 145952990 IC50 = 5 nM T59328 COA5Y3 145953378 IC50 > 1000 nM T59328 CN4Q7F 145953551 IC50 = 37 nM T59328 CT53JG 145953604 IC50 = 32 nM T59328 CMH8O2 145953998 IC50 = 34 nM T59328 C89RPH 145954372 IC50 > 1000 nM T59328 CBY18Z 145954422 IC50 = 32 nM T59328 CW2OE8 145954892 IC50 > 1000 nM T59328 CFB43Y 145956534 IC50 = 17 nM T59328 C5VSC7 145956704 IC50 = 5400 nM T59328 C2V8DA 145957160 IC50 > 1000 nM T59328 CA3E2C 145957992 IC50 = 162 nM T59328 C42ZQH 145958534 IC50 > 1000 nM T59328 CXWH23 145958592 IC50 > 1000 nM T59328 CJE35T 145958671 IC50 = 45.4 nM T59328 C2IHF1 145960158 IC50 = 3350 nM T59328 CV57UK 145960288 IC50 = 16.4 nM T59328 C9R0TU 145960317 IC50 = 240 nM T59328 CC7ZP1 145960400 IC50 = 1.7 nM T59328 C4D2AW 145962014 IC50 = 4.5 nM T59328 CJT41L 145962084 IC50 > 10000 nM T59328 C1R6UI 145963124 IC50 = 29 nM T59328 CICN74 145963796 IC50 = 16970 nM T59328 CRMN13 145963949 Ki = 1360 nM T59328 C9E0LZ 145964191 IC50 = 3900 nM T59328 C2JXB0 145964277 IC50 = 500 nM T59328 C4K6RY 145964618 IC50 = 100 nM T59328 CJYQ32 145964655 IC50 = 595.4 nM T59328 C0KJR5 145964906 IC50 = 650 nM T59328 CI52HO 145965123 IC50 = 675 nM T59328 CN41TJ 145965367 IC50 > 1000 nM T59328 CLM8E6 145965506 IC50 = 9350 nM T59328 C3ZD2W 145965608 IC50 = 3870 nM T59328 CI1UV7 145965620 Ki = 680 nM T59328 CO7IH0 145965741 IC50 = 940 nM T59328 CTQ9S5 145965923 IC50 = 6980 nM T59328 C7YM1B 145966210 IC50 = 31.8 nM T59328 CP2MX0 145966312 IC50 = 2400 nM T59328 C3YGN7 145966332 Ki = 810 nM T59328 CHY74R 145966422 Ki = 930 nM T59328 CZ38PG 145966502 Ki = 230 nM T59328 C8UWY5 145966767 IC50 = 78 nM T59328 C5L7VC 145966803 IC50 = 34.8 nM T59328 CQE9M5 145966810 IC50 > 10000 nM T59328 C0G8ED 145966828 IC50 > 1000000 nM T59328 C4LHS5 145967074 Ki = 140 nM T59328 C4OD9Q 145967187 IC50 = 1.3 nM T59328 CS7CR2 145967258 Ki = 164 nM T59328 CDW83M 145967332 IC50 = 267.6 nM T59328 COZA32 145967334 Ki = 170 nM T59328 CM41TV 145967355 IC50 = 82.6 nM T59328 CUE4K8 145967670 IC50 = 3.5 nM T59328 C7NJ9Q 145967774 IC50 = 2140 nM T59328 CDNC31 145967951 IC50 > 500 nM T59328 CA0IB1 145967983 IC50 = 22330 nM T59328 CJO79P 145968146 IC50 = 24.2 nM T59328 C5E8ZK 145968310 IC50 > 1000 nM T59328 CM7HI4 145968374 IC50 = 2.692 nM T59328 C6UAM8 145968450 IC50 = 1230 nM T59328 C4RX3Q 145968531 IC50 = 49 nM T59328 C8BH4I 145968555 IC50 = 3.2 nM T59328 CU5HJ8 145968616 IC50 = 4.2 nM T59328 C2J0VU 145968689 Ki = 2050 nM T59328 CHAU61 145968737 IC50 > 1000 nM T59328 C9IMB1 145968764 IC50 = 2.3 nM T59328 CWJ12M 145969155 IC50 > 10000 nM T59328 C2HN8R 145969194 IC50 > 1000 nM T59328 C0GDV8 145969399 IC50 = 249.1 nM T59328 C1N0GM 145969603 IC50 = 842.3 nM T59328 CK82QG 145969816 IC50 = 409 nM T59328 CVXS26 145969908 IC50 = 529 nM T59328 CX4C6R 145970163 IC50 = 270 nM T59328 CTD6N0 145970346 IC50 = 510 nM T59328 C9ZO3X 145970379 IC50 = 28 nM T59328 CXE6W9 145970478 IC50 = 3.9 nM T59328 C1C6YP 145970679 IC50 = 5.1 nM T59328 C8NK3O 145970839 IC50 = 596 nM T59328 CON74U 145970883 IC50 = 18 nM T59328 C8BKZ3 145971291 IC50 = 98 nM T59328 CQ4FP9 145971558 IC50 = 6020 nM T59328 CAV7I1 145971580 IC50 = 0.9 nM T59328 CSJ0X9 145971962 IC50 = 60 nM T59328 C5G7ZX 145972214 IC50 > 1000 nM T59328 CW8UY6 145972402 Ki = 330 nM T59328 CH18WC 145972585 IC50 = 5640 nM T59328 CVQP05 145972782 IC50 = 39 nM T59328 CKY02W 145972834 IC50 = 1160 nM T59328 CKQ46V 145972976 Ki = 110 nM T59328 CH5E2D 145973277 IC50 > 1000000 nM T59328 CM21LZ 145973281 IC50 > 1000 nM T59328 CWP85Z 145973302 IC50 > 1000 nM T59328 C64GAI 145973339 IC50 = 3250 nM T59328 CH5IM9 145973468 IC50 = 260 nM T59328 CFZX58 145973489 IC50 = 9760 nM T59328 CN6JG9 145973510 IC50 = 8070 nM T59328 CTPQ06 145973553 Ki = 2740 nM T59328 CIKF18 145973791 Ki = 320 nM T59328 CHGD35 145974340 IC50 = 72 nM T59328 CIWU86 145974353 Ki = 110 nM T59328 CQH3G7 145974613 IC50 = 1590 nM T59328 CXRY95 145974888 IC50 = 6900 nM T59328 C5JR6E 145974924 Ki = 2 nM T59328 CE35TV 145975018 IC50 = 1700 nM T59328 CX4S7R 145975100 IC50 = 9040 nM T59328 CI4JO0 145975282 IC50 = 0.9 nM T59328 C74TYP 145975351 IC50 > 100000 nM T59328 CSE6N1 145975386 IC50 = 190.6 nM T59328 C5HB7J 145975494 IC50 > 1000000 nM T59328 CZ98JF 145975496 IC50 = 1070 nM T59328 CCUX93 145975528 IC50 = 230 nM T59328 C2WK8V 145975646 IC50 = 2.1 nM T59328 C6MX1J 145976050 IC50 = 8550 nM T59328 C28GAM 145976336 IC50 = 1410 nM T59328 C3LR4O 145976442 IC50 = 2.4 nM T59328 C1IUN8 145976637 IC50 = 215.4 nM T59328 CI7S4L 145976764 Ki = 400 nM T59328 CH64BI 145976972 IC50 = 9970 nM T59328 CD82JO 145977064 IC50 = 3070 nM T59328 CG57KO 145977147 IC50 = 13 nM T59328 CX41WF 145977261 IC50 = 3800 nM T59328 C69INU 145977311 Ki = 3590 nM T59328 C7WZG3 145977617 IC50 = 14010 nM T59328 CMK7P9 145977756 Ki = 183 nM T59328 C15XGN 145977927 Ki = 80 nM T59328 C46QAV 145977992 Ki = 2520 nM T59328 C71TVY 145978029 IC50 = 51.9 nM T59328 C6JB8T 145978055 IC50 = 24.7 nM T59328 C81QRF 145978122 IC50 = 1.1 nM T59328 CXC9F7 145978377 IC50 = 900 nM T59328 CT1QE0 145978442 IC50 = 6070 nM T59328 C6JBH1 145978562 Ki = 940 nM T59328 CRCM82 145978681 IC50 = 51.3 nM T59328 C5IVB9 145978838 Ki = 161 nM T59328 CCT8N6 145978865 IC50 = 102 nM T59328 CM2NU5 145978997 IC50 = 15.3 nM T59328 CTA34O 145979089 IC50 = 23 nM T59328 C2D4CA 145979249 IC50 > 100 nM T59328 C5TP2U 145979643 IC50 = 45000 nM T59328 CE31VG 145979714 IC50 > 10000 nM T59328 CN7KH0 145979764 IC50 = 1.5 nM T59328 C4X8LC 145979928 IC50 > 1000000 nM T59328 CT9A2R 145980005 IC50 = 100.5 nM T59328 CV60SM 145980007 IC50 = 0.8 nM T59328 C9QFA1 145980052 IC50 = 21.4 nM T59328 CU05GX 145980058 IC50 = 0.7 nM T59328 CZEK06 145980063 IC50 = 3.2 nM T59328 C0P7JL 145980218 IC50 = 0.7 nM T59328 C4BM0U 145980284 IC50 = 22.4 nM T59328 CNFJ75 145980559 IC50 > 1000000 nM T59328 C5LIK2 145980611 IC50 = 1409 nM T59328 C1A5PW 145980662 IC50 = 27 nM T59328 CL19AW 145980663 IC50 = 0.4 nM T59328 CVRB57 145980676 IC50 = 0.6 nM T59328 COI8B7 145981029 IC50 = 9 nM T59328 C8FRT3 145981115 IC50 = 27 nM T59328 C4J9SC 145981182 IC50 = 105 nM T59328 CU67FB 145981262 IC50 = 2.7 nM T59328 C72RDL 145981281 IC50 = 46 nM T59328 CP67EO 145981349 IC50 = 68 nM T59328 CVO6T8 145981395 IC50 = 592.1 nM T59328 CSW6P0 145981487 IC50 = 1182 nM T59328 CCD7Y3 145981564 IC50 = 7200 nM T59328 C47TVC 145981655 IC50 = 1500 nM T59328 CLX91B 145981733 IC50 = 47.1 nM T59328 C64FYE 145981880 IC50 = 0.7 nM T59328 C1H5JE 145982613 IC50 = 52110 nM T59328 CC12YA 145982666 IC50 = 6.4 nM T59328 CF4BO8 145982785 IC50 = 4 nM T59328 CM6ZS7 145982824 IC50 = 3.1 nM T59328 CUN92A 145982933 IC50 = 21.5 nM T59328 C35FMR 145983116 IC50 > 100 nM T59328 C0YFS6 145983170 IC50 > 100 nM T59328 CF28AU 145983389 IC50 = 10.1 nM T59328 C48ZXP 145983545 IC50 > 100 nM T59328 C4QE7K 145983757 IC50 = 1200 nM T59328 CD5L8O 145983778 IC50 > 200 nM T59328 CM8Z7V 145984082 IC50 > 100 nM T59328 C1DM4I 145984486 IC50 = 1900 nM T59328 COPW70 145984516 IC50 = 1400 nM T59328 CYG42V 145984818 IC50 > 200 nM T59328 CLVN80 145984870 IC50 = 38730 nM T59328 CFS7D5 145984941 IC50 > 200 nM T59328 C05IMJ 145984942 IC50 = 7.1 nM T59328 CPHN84 145985403 IC50 = 467 nM T59328 CS9C8J 145986155 IC50 > 200 nM T59328 CY5NX4 145986312 IC50 = 1 nM T59328 C2T4PK 145986404 IC50 = 5600 nM T59328 CV45JH 145986520 IC50 = 754 nM T59328 C8EUL5 145986728 IC50 = 2700 nM T59328 CB80EO 145986808 IC50 > 1000 nM T59328 CCJ19R 145986823 IC50 = 2.6 nM T59328 CGI48S 145986878 IC50 = 0.3 nM T59328 CB48CA 145986981 IC50 = 0.7 nM T59328 C1Y5MO 145987062 IC50 = 632.8 nM T59328 CRKD41 145987099 IC50 = 901 nM T59328 CAE5G0 145987157 IC50 > 1000000 nM T59328 CJ2A5I 145987445 IC50 = 951 nM T59328 CU96RK 145987761 IC50 = 944 nM T59328 CF6KO7 145987807 IC50 = 1 nM T59328 C0MI7K 145988025 IC50 = 21 nM T59328 C7A4WK 145988274 IC50 = 47.7 nM T59328 C3N8OJ 145988373 IC50 = 288 nM T59328 C4FWV5 145988395 IC50 = 1931 nM T59328 CDVL79 145988898 IC50 = 33 nM T59328 CZ1VH0 145988939 IC50 = 94.7 nM T59328 C9BX4U 145988956 IC50 > 10000 nM T59328 CP9N1M 145989301 IC50 = 205 nM T59328 C74MSY 145989401 IC50 = 17 nM T59328 C2VA1T 145989472 IC50 = 1700 nM T59328 C2B0LS 145989721 IC50 = 62.5 nM T59328 CB13UV 145989878 IC50 = 0.8 nM T59328 CWI75O 145990017 IC50 = 120 nM T59328 C2PBJ5 145990245 IC50 = 112 nM T59328 CH17ZV 145990291 IC50 = 13.4 nM T59328 CX4YJ5 145990338 IC50 = 0.71 nM T59328 CTC0L2 145990413 IC50 = 60 nM T59328 CE1QB4 145990507 IC50 = 229 nM T59328 CNQ91H 145990537 IC50 = 26 nM T59328 C9Q6XC 145990684 IC50 = 0.7 nM T59328 COS6Z7 145990801 IC50 = 24.8 nM T59328 C1J5IX 145990848 IC50 > 1000000 nM T59328 CRS5P2 145991103 IC50 = 1.4 nM T59328 CD79LS 145991130 IC50 = 9800 nM T59328 C0XBV2 145991309 IC50 = 752 nM T59328 C5KB0A 145991472 IC50 > 1000000 nM T59328 COU0E6 145991881 IC50 = 91.7 nM T59328 C2CBQ4 145992100 IC50 = 751 nM T59328 C4YUL3 145992531 IC50 = 96.6 nM T59328 CZP7Y0 145992597 IC50 = 1229 nM T59328 C4A2UC 145992646 IC50 = 70 nM T59328 C2FQG8 145992679 IC50 = 2800 nM T59328 CO41PW 145992706 IC50 = 792 nM T59328 CNC69T 145992844 IC50 > 100000 nM T59328 C0C4ZD 145993006 IC50 = 11 nM T59328 CWK20P 145993042 IC50 = 108 nM T59328 C7Q6NU 145993198 IC50 = 933 nM T59328 CW8E2A 145993359 IC50 = 1 nM T59328 C85KQX 145993400 IC50 = 1.2 nM T59328 CZ6OC9 145993414 IC50 = 37 nM T59328 CS8UQ5 145994037 IC50 = 8.6 nM T59328 C6B3TD 146014465 IC50 = 13 nM T59328 CQNH23 146180715 IC50 = 9.3 nM T59328 C6YC0B 146180716 IC50 = 179.6 nM T59328 CJU8M7 146180717 IC50 = 2.2 nM T59328 CS6FR4 146180753 IC50 = 19.2 nM T59328 CK18RY 146180803 IC50 = 37.1 nM T59328 CS2Q4N 146182117 IC50 = 7.9 nM T59328 CF06AW 146197277 IC50 > 20000 nM T59328 CRP36X 146197294 IC50 > 20000 nM T59328 COJM12 146197324 IC50 > 20000 nM T59328 C8S7QZ 146197334 IC50 > 20000 nM T59328 C9MO7E 146197361 IC50 > 20000 nM T59328 CW9Y5K 146197370 IC50 > 20000 nM T59328 CO27GX 146197371 IC50 > 20000 nM T59328 CFV2O7 146197389 IC50 > 20000 nM T59328 C1X2MP 146197393 IC50 > 20000 nM T59328 C0CN9F 146197408 IC50 > 20000 nM T59328 CO1F2N 146197447 IC50 > 20000 nM T59328 CBJR67 146197457 IC50 > 20000 nM T59328 CG86IF 146197468 IC50 > 20000 nM T59328 CD7Y8E 146212989 IC50 > 20000 nM T59328 CBM7C5 146773032 IC50 = 12450 nM T59328 CP81CX 146832100 IC50 = 76 nM T59328 C9D1EH 147117461 IC50 = 18690 nM T59328 C8I1HV 147384518 IC50 = 16180 nM T59328 C7DYK4 147709549 IC50 = 18260 nM T59328 CIT79C 148291912 IC50 = 9570 nM T59328 C2U0SJ 148390225 IC50 = 26970 nM T59328 CJ23ZE 148637488 IC50 = 15360 nM T59328 CVL49H 149513019 IC50 = 22850 nM T59328 CR20QN 149611945 IC50 = 39 nM T59328 CYN8L2 152157601 IC50 > 10000 nM T59328 CSE96B 152685456 IC50 = 315 nM T59328 CFKU39 152790957 IC50 = 30450 nM T59328 CS7Q1E 152878273 IC50 = 52 nM T59328 CV41DF 153011787 IC50 = 25410 nM T59328 C60JPV 155166360 IC50 = 149 nM T59328 CL41OU 155183985 IC50 = 2 nM T59328 C90HPT 155338585 IC50 = 31 nM T59328 CP5NX6 155338590 IC50 = 12 nM T59328 CRC8D2 155489850 IC50 = 2200 nM T59328 CZ4V5U 155510439 IC50 > 1000 nM T59328 C03YFP 155510706 IC50 = 38 nM T59328 C5Z7GK 155511049 IC50 = 4.95 nM T59328 CDR04S 155511317 IC50 = 15 nM T59328 CQI50K 155511379 IC50 = 81 nM T59328 CY7X0V 155511571 IC50 = 28.2 nM T59328 CWZ2S8 155511862 IC50 = 4.3 nM T59328 CE10PX 155512047 IC50 = 5 nM T59328 CL4B2M 155512535 IC50 = 147 nM T59328 CKR0P6 155512805 IC50 = 25 nM T59328 C81YCJ 155513061 IC50 = 70 nM T59328 C9NT2X 155513114 IC50 = 30 nM T59328 C2MD1Q 155513187 IC50 > 10000 nM T59328 CQ3XH4 155513485 IC50 = 500 nM T59328 COZ61S 155513553 IC50 = 46.52 nM T59328 CU12GD 155513666 IC50 = 10580 nM T59328 C17INE 155513714 IC50 = 397 nM T59328 CI78ZM 155513927 IC50 = 10 nM T59328 C7SK0E 155513959 IC50 = 40.6 nM T59328 C1XNV5 155513991 IC50 = 9 nM T59328 CHG6K2 155514100 IC50 = 320 nM T59328 CBP9L6 155514128 IC50 = 450 nM T59328 CKN04R 155514224 IC50 = 34 nM T59328 C3EXJ1 155514609 IC50 = 52.6 nM T59328 C7SPR0 155514679 IC50 = 111 nM T59328 CD46IN 155514865 IC50 = 61 nM T59328 C7YEN3 155514902 IC50 = 0.87 nM T59328 C7AMX8 155514903 IC50 > 3000 nM T59328 C1K3OA 155515133 IC50 = 710 nM T59328 CDAL34 155515494 IC50 = 844 nM T59328 CT2C5D 155515585 IC50 = 54.69 nM T59328 CC7N4A 155515743 IC50 = 4520 nM T59328 CU76NE 155516227 IC50 = 24130 nM T59328 CI23DH 155516489 IC50 = 1257 nM T59328 CR2D9I 155516959 IC50 = 16 nM T59328 C8GX0B 155517202 IC50 = 2700 nM T59328 C4D1WA 155517369 IC50 = 4750 nM T59328 C36ZMS 155518518 IC50 > 50000 nM T59328 C86HPW 155518524 IC50 = 10000 nM T59328 CJ0O8S 155518727 IC50 = 1248 nM T59328 CPTF82 155518915 IC50 = 79 nM T59328 CH42VE 155518994 IC50 = 2459 nM T59328 CG4C2D 155519085 IC50 = 500 nM T59328 C3VTM7 155519139 IC50 = 400 nM T59328 C0BZ6I 155519249 IC50 = 416 nM T59328 CTS0J7 155519458 IC50 = 400 nM T59328 CE83DJ 155519522 IC50 = 1259 nM T59328 C3NA2I 155519537 IC50 > 1000 nM T59328 CC8BO2 155519579 IC50 = 1700 nM T59328 CR68FM 155519610 IC50 > 1000 nM T59328 C9HEY1 155519702 IC50 = 26150 nM T59328 CYO23E 155519705 IC50 = 32.5 nM T59328 CBY13X 155519739 EC50 = 2 nM T59328 CNU28S 155519814 IC50 > 1000 nM T59328 CQAN74 155519895 IC50 = 105 nM T59328 C01HMD 155519991 IC50 = 239 nM T59328 C1X6YD 155520212 IC50 = 1322 nM T59328 C6K8NG 155520384 IC50 = 499 nM T59328 COQ7U0 155520571 EC50 = 4 nM T59328 C98UXO 155520734 IC50 = 0.34 nM T59328 C3UAF7 155521257 IC50 = 65.34 nM T59328 C9FVT0 155521452 IC50 = 123.2 nM T59328 CF93WQ 155521654 IC50 = 395 nM T59328 CWVX73 155522179 IC50 = 54.99 nM T59328 C8ZDA3 155522205 IC50 = 562 nM T59328 CNIR83 155522516 IC50 = 224.1 nM T59328 CB50GK 155522849 IC50 = 43.56 nM T59328 CHRT30 155522905 IC50 = 20 nM T59328 CI65WG 155523218 IC50 = 227.9 nM T59328 CES5L2 155523448 IC50 = 65.2 nM T59328 CNLC48 155523465 IC50 = 23.4 nM T59328 C2NQV1 155523617 IC50 = 421 nM T59328 CZ6ES5 155524096 IC50 = 0.5872 nM T59328 CA9YF3 155524153 IC50 = 38 nM T59328 C5EZR1 155524215 IC50 = 68 nM T59328 CD7ZH8 155524226 IC50 > 20000 nM T59328 C3TF9E 155524436 IC50 = 120.7 nM T59328 C5R8SL 155524645 IC50 > 20000 nM T59328 CH6FQ9 155524667 IC50 = 4300 nM T59328 CJBE61 155524820 IC50 = 6300 nM T59328 C0COA7 155525819 IC50 = 62 nM T59328 CJ35GA 155525934 IC50 = 4240 nM T59328 CRT67D 155526236 IC50 = 8.7 nM T59328 CFAS17 155526847 IC50 = 13 nM T59328 CE3OH1 155527121 IC50 = 138 nM T59328 C3GNP6 155527669 IC50 = 2.5 nM T59328 C8I3SW 155527677 IC50 = 12 nM T59328 CQLF39 155527847 IC50 = 16.43 nM T59328 C3HP8E 155527851 IC50 = 18 nM T59328 CF39US 155528086 IC50 = 421 nM T59328 C72HJM 155528259 IC50 > 1000 nM T59328 C47YUC 155528358 IC50 > 20000 nM T59328 C9P2NQ 155528441 IC50 = 8770 nM T59328 CHI54P 155529236 IC50 = 617 nM T59328 C10JWF 155529388 IC50 = 14 nM T59328 CFKV53 155529663 IC50 = 22.7 nM T59328 CW9OC4 155529736 IC50 = 37.1 nM T59328 CN40AE 155529739 IC50 = 700 nM T59328 CUXA18 155529935 IC50 = 903 nM T59328 CLJ5T9 155529954 IC50 = 18.54 nM T59328 CU96GQ 155529955 IC50 = 64 nM T59328 CL0US4 155530459 IC50 = 2.3 nM T59328 CQLV68 155530541 IC50 = 1600 nM T59328 C6VQ0W 155530641 IC50 > 1000 nM T59328 C2WCU6 155530774 IC50 = 1048 nM T59328 C3N4UG 155530777 IC50 = 1771 nM T59328 CX7I1V 155531079 IC50 = 765 nM T59328 CWO98B 155531773 IC50 = 9 nM T59328 CVBK76 155531967 IC50 > 1000 nM T59328 C8HDO1 155532442 IC50 = 3 nM T59328 CGVZ73 155532854 IC50 > 1000 nM T59328 C3D5JZ 155533027 IC50 = 177 nM T59328 CJ6T5H 155533092 IC50 = 12 nM T59328 CNQP76 155533136 IC50 > 1000 nM T59328 CQFC65 155533189 IC50 = 2400 nM T59328 C7OX2W 155533223 IC50 = 19.97 nM T59328 CNGX84 155533637 IC50 = 2750 nM T59328 C5UQG3 155534199 IC50 = 8.7 nM T59328 C1NGV5 155534208 IC50 = 499 nM T59328 C4TRF0 155534357 IC50 = 3660 nM T59328 C3J4OM 155534528 IC50 > 20000 nM T59328 CM0U3I 155534552 IC50 > 1000 nM T59328 CEQJ52 155534874 IC50 > 1000 nM T59328 C6QX2V 155534940 IC50 = 31.7 nM T59328 CMH2J4 155535076 IC50 = 0.69 nM T59328 CD8TO7 155535214 IC50 = 15330 nM T59328 C3RWB0 155535296 IC50 = 31 nM T59328 CRI7V1 155535998 IC50 = 1753 nM T59328 C78MZC 155536330 IC50 = 2 nM T59328 C6H7QE 155536433 IC50 = 83 nM T59328 CF0A9O 155536643 IC50 = 10 nM T59328 CBS75N 155536946 IC50 = 2800 nM T59328 C2CG1A 155537016 IC50 > 10000 nM T59328 C2SW1K 155537706 IC50 = 201 nM T59328 CP3AD2 155537718 IC50 = 81 nM T59328 CZNX25 155537733 IC50 = 234 nM T59328 CP8ZV6 155538283 IC50 = 4 nM T59328 C6Z7XO 155538664 IC50 = 2.213 nM T59328 C0IH1J 155539209 IC50 = 105.3 nM T59328 CEN71T 155539953 IC50 = 20.83 nM T59328 CC3IQ7 155540048 IC50 = 26 nM T59328 C1B0VO 155540273 IC50 = 4.3 nM T59328 CE46SL 155540854 IC50 = 4340 nM T59328 C5O4JM 155540856 IC50 = 23340 nM T59328 CX68YN 155541385 IC50 > 50000 nM T59328 CLY07P 155541605 IC50 > 150 nM T59328 CT02GE 155541767 IC50 = 598 nM T59328 CH10DU 155542091 IC50 = 654 nM T59328 CNR2X9 155542138 IC50 = 119.7 nM T59328 C7X2KJ 155542371 IC50 = 70 nM T59328 CP67JN 155542393 IC50 = 5.9 nM T59328 C02VLJ 155542715 IC50 = 4 nM T59328 CTQ9S4 155543012 IC50 = 1.4 nM T59328 CW73EO 155543439 IC50 = 38 nM T59328 C1VJH0 155543634 IC50 = 36840 nM T59328 C0JR1M 155544107 IC50 = 0.62 nM T59328 CUT37P 155544297 IC50 = 20 nM T59328 C5ZMA0 155544307 IC50 = 5004 nM T59328 CVG79N 155544855 IC50 = 3059 nM T59328 C1SMF6 155545153 IC50 = 133 nM T59328 CGE04I 155545288 IC50 = 820 nM T59328 CEJ3V2 155545290 IC50 = 56.1 nM T59328 C4H9XV 155545331 IC50 = 209 nM T59328 CCHK04 155545559 IC50 = 50.8 nM T59328 CPKS19 155545810 IC50 = 5 nM T59328 CN18UI 155545963 IC50 = 14 nM T59328 C46MQV 155546345 IC50 = 9 nM T59328 CJN15V 155546412 IC50 = 6.24 nM T59328 CSI83K 155546458 IC50 = 12.93 nM T59328 CAVB85 155546598 IC50 > 10000 nM T59328 CTBA51 155546884 IC50 = 6 nM T59328 CFA1X6 155546954 IC50 = 6.6 nM T59328 C10XPU 155547167 EC50 = 666 nM T59328 CN4PM8 155547174 IC50 = 1.15 nM T59328 C7SF2C 155547229 IC50 > 10000 nM T59328 CL8X7V 155547722 IC50 = 48.07 nM T59328 CFR63D 155547749 IC50 = 275.7 nM T59328 CGX7Z0 155548089 IC50 = 40 nM T59328 C60YKA 155548301 IC50 > 1000 nM T59328 CV54FM 155548416 IC50 = 6600 nM T59328 CE6M4K 155548572 IC50 = 174 nM T59328 CBN4M1 155548812 IC50 = 44 nM T59328 CZ7WR0 155549232 IC50 = 8 nM T59328 CNG4O3 155549841 IC50 = 2900 nM T59328 CL1E6U 155549934 IC50 = 27.92 nM T59328 CY6RU2 155549975 IC50 = 0.37 nM T59328 CV7S6N 155550199 IC50 = 4 nM T59328 C9J1MU 155550347 IC50 = 2 nM T59328 C93NWJ 155550657 IC50 = 148.8 nM T59328 C49SQG 155551406 IC50 = 23 nM T59328 C3UBY1 155551683 IC50 = 1128.9 nM T59328 CEDT28 155552106 IC50 = 26 nM T59328 CZ4J2P 155552610 IC50 > 1000 nM T59328 C0HUL3 155552710 IC50 = 1975 nM T59328 C2VNW3 155553566 IC50 = 52 nM T59328 CAC31S 155553712 IC50 = 2 nM T59328 CGVU70 155554426 IC50 = 4710 nM T59328 C5MAK6 155554594 IC50 = 45.2 nM T59328 CJ0G2I 155554715 IC50 = 35 nM T59328 CD9M1F 155554777 IC50 = 273 nM T59328 C2T1XS 155554878 IC50 = 591 nM T59328 C1FJ5D 155555800 IC50 > 20000 nM T59328 CT6S9X 155555827 IC50 = 120.2 nM T59328 CWDR07 155555935 IC50 = 15630 nM T59328 C3F8YQ 155556804 IC50 = 368 nM T59328 CX96CQ 155556857 IC50 = 32.61 nM T59328 C5KSJ1 155556978 IC50 = 93 nM T59328 C4BH8P 155557234 IC50 = 12 nM T59328 CQ9GK2 155557533 IC50 = 27 nM T59328 C2LWI3 155557949 IC50 = 157 nM T59328 CARD46 155557959 IC50 = 197 nM T59328 CZD71I 155558249 IC50 = 3.11 nM T59328 CC8R3X 155558455 IC50 = 188 nM T59328 C10OFJ 155558962 IC50 = 0.6 nM T59328 CPAV79 155559005 IC50 > 3000 nM T59328 C89XOB 155559201 IC50 = 5.6 nM T59328 C2Q8OK 155559257 IC50 = 105 nM T59328 CL3JM7 155559534 IC50 = 153.5 nM T59328 C1OI5K 155559863 IC50 > 1000 nM T59328 CBA35K 155559950 IC50 = 77 nM T59328 C51IBQ 155560019 IC50 = 937 nM T59328 CXZ74V 155560104 IC50 > 150 nM T59328 CCD34P 155560610 IC50 = 3200 nM T59328 CT2XQ0 155561007 IC50 = 215 nM T59328 C8J0IZ 155561310 IC50 > 1000 nM T59328 CM3JG6 155561359 IC50 = 2 nM T59328 C6N1KS 155561750 IC50 = 146.2 nM T59328 CES3Q5 155561884 IC50 = 1200 nM T59328 CT7UJ9 155562064 IC50 = 104 nM T59328 CFI4C8 155562148 IC50 = 85 nM T59328 CC5F3I 155562216 IC50 = 84 nM T59328 CTF4Z2 155562466 IC50 > 1000 nM T59328 C87PUX 155562472 IC50 = 107.2 nM T59328 CNDL07 155562495 IC50 = 141 nM T59328 C1VCU9 155562538 IC50 = 33.31 nM T59328 C1ZX4J 155563060 IC50 > 1000 nM T59328 C9V5HT 155563732 IC50 = 142.7 nM T59328 C9L6WZ 155563761 IC50 > 150 nM T59328 C7XK2B 155564005 IC50 = 118.6 nM T59328 CS37KE 155564015 IC50 = 12000 nM T59328 CAC85T 155564156 IC50 > 3000 nM T59328 CT53XC 155564242 IC50 = 1 nM T59328 CU7Z0H 155564272 IC50 = 3.7 nM T59328 CLPY65 155564381 IC50 = 326 nM T59328 CY9BN3 155564537 IC50 = 11 nM T59328 C3F6ML 155564606 IC50 = 2160 nM T59328 CQ1N7J 155564622 IC50 = 38.5 nM T59328 CY1KP0 155564719 IC50 = 92 nM T59328 CBS5F3 155564756 IC50 = 8 nM T59328 C0ZWD9 155565268 IC50 = 302 nM T59328 C0UG5P 155565835 IC50 > 150 nM T59328 CA36ST 155565961 IC50 = 19 nM T59328 CWAF51 155566440 IC50 = 12 nM T59328 C3G5LQ 155566848 IC50 > 1000 nM T59328 C04KYS 155566973 IC50 = 8.3 nM T59328 CZC73X 155567166 IC50 = 2880 nM T59328 CUB2J0 155567333 IC50 = 1400 nM T59328 C5AO3Q 155567359 IC50 = 60 nM T59328 C6LI4S 155567410 IC50 = 12.57 nM T59328 CQS81I 155568841 IC50 = 108 nM T59328 CMNZ49 155569055 IC50 > 2000 nM T59328 CGU74Q 155569301 IC50 = 150 nM T59328 C1IC3A 14862543 IC50 = 40000 nM T59328 CLQ6F4 14862545 IC50 = 7000 nM T59328 D00ATA 5908088 IC50 > 100000 nM T59328 D00ERW 44444843 Ki > 1803 nM T59328 D00GVV 5329155 IC50 > 100000 nM T59328 D00HVA 11624601 Ki > 1800 nM T59328 D00LRC 10422592 IC50 > 20000 nM T59328 D00RBV 10445611 IC50 > 25000 nM T59328 D00RIX 5280443 IC50 = 30 ug.mL-1 T59328 D00TBD 10461815 IC50 = 3800 nM T59328 D00TJF 11807783 IC50 = 3.38 nM T59328 D00TZD 2776 IC50 = 0.37 nM T59328 D00VZA 5328763 IC50 = 1000 nM T59328 D00WZG 44442168 IC50 = 15 nM T59328 D01NTW 5328768 Ki = 3500 nM T59328 D01OKF 46207013 IC50 = 580 nM T59328 D01RHR 71519693 IC50 = 11 nM T59328 D01UYS 11778521 IC50 > 20000 nM T59328 D01VFR 4708 IC50 = 0.08 nM T59328 D01WXV 44442181 IC50 = 15 nM T59328 D01WYI 9995195 IC50 = 0.42 nM T59328 D02BUW 2061 Ki = 1000 nM T59328 D02BXJ 46864270 IC50 = 736 nM T59328 D02CUF 10424517 IC50 > 20000 nM T59328 D02KVB 5328804 IC50 = 125 nM T59328 D02NNT 53232451 IC50 > 10000 nM T59328 D02RIG 5328755 IC50 = 7000 nM T59328 D02ZRO 735125 IC50 = 27 nM T59328 D03ATU 4707 IC50 = 0.008 nM T59328 D03BJB 9549299 IC50 = 21 nM T59328 D03CVQ 44442182 IC50 = 5 nM T59328 D03EHM 24905142 IC50 = 260 nM T59328 D03HLH 44331231 IC50 = 70 nM T59328 D03MUZ 17759555 IC50 = 1800 nM T59328 D03OKV 9844320 IC50 > 1000 nM T59328 D03XDN 4709 IC50 = 0.1 nM T59328 D04FNY 25195216 IC50 = 3480 nM T59328 D04HGN 2809539 IC50 = 6300 nM T59328 D04LXG 44442183 IC50 = 140 nM T59328 D04NGS 5330790 IC50 > 100000 nM T59328 D04PEI 11467730 IC50 > 50000 nM T59328 D04XNJ 4879 IC50 = 2700 nM T59328 D05ARF 5328077 IC50 = 578 nM T59328 D05EDW 10085862 IC50 > 20000 nM T59328 D05FFT 11566580 IC50 = 0.3 nM T59328 D05GBY 10242258 IC50 > 20000 nM T59328 D05QMN 44331083 IC50 = 2500 nM T59328 D05SNG 10398928 IC50 > 20000 nM T59328 D06BJG 71556703 IC50 = 7 nM T59328 D06HVH 54613583 IC50 > 10000 nM T59328 D06KSF 9549300 IC50 < 5000 nM T59328 D06LJL 9916282 IC50 = 800 nM T59328 D06LLF 10017166 IC50 > 20000 nM T59328 D06MCJ 9972296 IC50 > 20000 nM T59328 D06QWO 14824655 IC50 > 10 ug.mL-1 T59328 D06UEK 15984068 IC50 = 710 nM T59328 D06VNR 10085863 IC50 > 20000 nM T59328 D07CFT 10447210 IC50 > 20000 nM T59328 D07IHD 5328753 IC50 = 500 nM T59328 D07IHM 9823787 IC50 > 10000 nM T59328 D07JDY 10243001 IC50 > 20000 nM T59328 D07OCA 5330812 IC50 > 10000 nM T59328 D07OSK 6419834 IC50 > 100000 nM T59328 D07OXC 11650194 IC50 = 1700 nM T59328 D07SRX 9797919 IC50 = 7300 nM T59328 D07UYV 2857 IC50 = 0.006 nM T59328 D07ZWN 10060170 IC50 > 20000 nM T59328 D08JGS 11722903 IC50 > 20000 nM T59328 D08KWL 10402251 IC50 > 20000 nM T59328 D08LYB 5166 IC50 = 83 nM T59328 D08NQM 5289247 IC50 > 10000 nM T59328 D08RZB 11153014 IC50 = 5200 nM T59328 D08SUH 10336427 IC50 > 20000 nM T59328 D08WOG 9948853 IC50 = 20 nM T59328 D09HVH 135566652 IC50 > 10 nM T59328 D09LPL 5329103 IC50 = 3000 nM T59328 D09QBA 23378546 IC50 > 10000 nM T59328 D09TNR 9850161 IC50 > 10000 nM T59328 D09XIL 11396738 IC50 = 545 nM T59328 D0A0JL 2052 Ki = 11000 nM T59328 D0A1CM 5281855 IC50 = 690 nM T59328 D0A4XJ 5289418 IC50 > 100000 nM T59328 D0A6AA 10083695 IC50 > 20000 nM T59328 D0A6YP 9971060 IC50 > 20000 nM T59328 D0A9RM 5281804 IC50 = 4 ug.mL-1 T59328 D0AO6T 10402592 IC50 > 20000 nM T59328 D0AU0M 637542 Ki = 1000000 nM T59328 D0B4PH 2426 IC50 = 0.12 nM T59328 D0B8DE 135469328 IC50 = 5000 nM T59328 D0BU6T 354471 IC50 = 500 nM T59328 D0BW4G 10907042 IC50 > 30000 nM T59328 D0C1BE 10401378 IC50 > 20000 nM T59328 D0C2GE 67161540 IC50 = 137 nM T59328 D0C9KC 10850934 IC50 = 95 nM T59328 D0CF9B 10265642 IC50 > 20000 nM T59328 D0D2FC 2794188 IC50 = 5100 nM T59328 D0D5EW 5311104 IC50 = 390 nM T59328 D0D6DH 10125830 IC50 > 50000 nM T59328 D0D6MH 11617559 IC50 > 24000 nM T59328 D0D9PD 11656591 IC50 = 720 nM T59328 D0D9TU 3894 IC50 = 0.004 ug.mL-1 T59328 D0DF3Z 2808977 IC50 = 4.6 nM T59328 D0EE6A 6398883 IC50 > 1000 nM T59328 D0EH6L 10360970 IC50 = 4500 nM T59328 D0EU1R 46215815 IC50 > 10000 nM T59328 D0EW3L 5281222 IC50 = 8000 nM T59328 D0F6FZ 10494722 IC50 = 90 nM T59328 D0FH3M 18770833 IC50 = 4000 nM T59328 D0G0KN 9882618 IC50 > 20000 nM T59328 D0G0ZQ 10468421 IC50 > 20000 nM T59328 D0G3SZ 6918469 IC50 = 9.8 ug.mL-1 T59328 D0G3TK 5280863 IC50 = 3 ug.mL-1 T59328 D0G4HR 14862522 IC50 = 1000 nM T59328 D0G6SA 10422972 IC50 > 20000 nM T59328 D0G8GA 350901 IC50 = 15000 nM T59328 D0G9KD 5328245 IC50 = 0.003 nM T59328 D0GN3E 10243546 IC50 > 20000 nM T59328 D0GW4Q 5330524 IC50 = 380 nM T59328 D0H2CM 135565635 IC50 = 4400 nM T59328 D0H3UI 2063 Ki > 400000 nM T59328 D0H4JB 11778467 IC50 > 20000 nM T59328 D0HD2G 4788 IC50 = 25000000 nM T59328 D0HE0E 5941540 IC50 > 100000 nM T59328 D0HM5W 5328042 IC50 = 0.78 nM T59328 D0I0GL 10039460 IC50 > 20000 nM T59328 D0I7RA 11696664 IC50 = 131 nM T59328 D0IR5I 135453851 IC50 = 500 nM T59328 D0J5SK 5328819 IC50 = 2700 nM T59328 D0K2VO 44442165 IC50 = 14 nM T59328 D0K7GD 5328045 IC50 = 0.1 nM T59328 D0K9ON 10040402 IC50 > 20000 nM T59328 D0KF3N 10083699 IC50 > 20000 nM T59328 D0L0HG 766949 IC50 > 10000 nM T59328 D0L3FK 5289419 IC50 > 10000 nM T59328 D0L3SN 6439158 IC50 = 8800 nM T59328 D0L4HJ 5330462 IC50 = 5400 nM T59328 D0L8HO 2399 IC50 > 50000 nM T59328 D0M4SY 135440466 IC50 = 1600 nM T59328 D0M9QM 5327820 IC50 = 800 nM T59328 D0ME9B 46868971 IC50 > 10 nM T59328 D0N8TQ 10401956 IC50 < 1 nM T59328 D0NH7M 5328760 IC50 = 370 nM T59328 D0NS1S 5280442 IC50 = 40 ug.mL-1 T59328 D0O6OH 71553154 IC50 = 590 nM T59328 D0O9UR 638439 IC50 = 7900 nM T59328 D0P0RD 10065445 IC50 > 20000 nM T59328 D0P0WT 3139 IC50 > 10000 nM T59328 D0P2GE 18770812 IC50 = 5600 nM T59328 D0P3JW 447700 IC50 = 90 nM T59328 D0P6JS 11675054 IC50 > 10000 nM T59328 D0Q0YV 24944925 IC50 > 19952.62 nM T59328 D0Q3EW 9549303 IC50 > 10000 nM T59328 D0Q3GG 667601 Ki = 850 nM T59328 D0Q3NG 11715520 Ki > 1800 nM T59328 D0QC0W 9914412 IC50 = 110 nM T59328 D0QN6U 9806182 IC50 > 10000 nM T59328 D0RD5S 10355832 IC50 > 20000 nM T59328 D0S0RK 10680 IC50 = 50 ug.mL-1 T59328 D0S7IE 11658882 Ki > 1800 nM T59328 D0S9QP 44442180 IC50 = 26 nM T59328 D0S9YX 5280373 IC50 = 30 ug.mL-1 T59328 D0SJ2Q 10494 IC50 > 20000 nM T59328 D0SY2M 5281708 IC50 > 100 ug.mL-1 T59328 D0T9FQ 10061448 IC50 > 10000 nM T59328 D0U3WQ 9817165 IC50 > 30000 nM T59328 D0U6WB 2427 IC50 = 0.025 nM T59328 D0UN9O 3385203 IC50 >= 10000 nM T59328 D0V8QI 10331922 IC50 > 20000 nM T59328 D0V9EN 689043 Ki = 400000 nM T59328 D0W1BE 638437 IC50 = 10000 nM T59328 D0W6CE 10644450 IC50 = 10500 nM T59328 D0W7IN 10083051 IC50 > 20000 nM T59328 D0W9BF 9903563 IC50 > 20000 nM T59328 D0WW8M 10446889 IC50 > 20000 nM T59328 D0X4IO 5350 IC50 = 9000 nM T59328 D0X4UE 10220590 IC50 = 1000 nM T59328 D0XS9E 5330535 IC50 > 30000 nM T59328 D0Y2AM 5328038 IC50 = 355 nM T59328 D0YE1X 9927943 IC50 > 10000 nM T59328 D0YZ7H 9797370 IC50 > 100000 nM T59328 D0Z4HV 10354294 IC50 > 10000 nM T59328 D0Z7TM 22273644 IC50 > 1000 nM T59328 D0ZH1U 2051 IC50 = 120 nM T59328 D0ZT9D 6450172 IC50 = 1600 nM T91959 D06NVJ 936 IC50 = 30000 nM T91959 D0E3SH 6918837 Ki > 10000 nM T91959 D09XIZ 11538455 Ki > 10000 nM T91959 D0E3LP 5113032 IC50 = 48700 nM T91959 D0U3EP 445154 EC50 > 300000 nM T91959 D04JZE 3246390 IC50 = 12900 nM T91959 CPQ82T 95692 IC50 = 23000 nM T91959 CJ7U9O 96455 IC50 = 235000 nM T91959 CLY6K3 661302 IC50 > 100000 nM T91959 CBD84H 698853 IC50 = 29300 nM T91959 C0XD3L 1096276 IC50 > 100000 nM T91959 C1RVS5 1096292 IC50 > 100000 nM T91959 C6YS9Z 1103548 IC50 = 46400 nM T91959 CE4KD6 1142691 IC50 = 116300 nM T91959 CPI3Q1 1183101 IC50 > 50000 nM T91959 CU7ZT4 1183103 IC50 > 50000 nM T91959 CUJ7W0 1183104 IC50 > 50000 nM T91959 CLK57R 1183106 IC50 > 50000 nM T91959 CH9V7F 1183108 IC50 > 50000 nM T91959 CC8V0S 1328033 IC50 > 50000 nM T91959 CB7I9R 1372572 IC50 > 5000 nM T91959 CB92ZQ 1372991 IC50 = 30300 nM T91959 C4JD2N 2130402 IC50 > 50000 nM T91959 C94ELI 3610426 IC50 = 40300 nM T91959 CJ0T4E 3612016 IC50 > 100000 nM T91959 CN8F1I 3953303 IC50 > 50000 nM T91959 CQ25OP 9833992 IC50 = 38000 nM T91959 CL2VP6 24180124 EC50 > 300000 nM T91959 CL4WV2 24180125 IC50 = 850 nM T91959 CQI29M 24180126 EC50 > 300000 nM T91959 CI1R0Y 24772043 IC50 = 25700 nM T91959 CCQ1R9 44138532 IC50 > 300000 nM T91959 C6L5KB 45168044 IC50 > 100000 nM T91959 C52OHP 45483031 IC50 > 100000 nM T91959 C67ICN 45486324 IC50 = 24000 nM T91959 CMF17W 46871954 IC50 = 4500 nM T91959 C4B0WG 46871955 IC50 = 4300 nM T91959 CU64YT 53379498 IC50 = 57200 nM T91959 C3T8YQ 56664966 IC50 = 213500 nM T91959 CC7T2A 56674921 IC50 = 25100 nM T91959 CZ25SN 56935695 IC50 > 300000 nM T91959 C92ZDR 59053311 IC50 = 540 nM T91959 CE4IP3 60141294 IC50 > 200000 nM T91959 CM08ZL 60148504 IC50 > 300000 nM T91959 C94IGH 66560391 IC50 > 200000 nM T91959 CNVG06 71304813 IC50 = 4 nM T91959 CWY4S0 71304814 IC50 = 33 nM T91959 C4BHW5 71304815 IC50 = 7.2 nM T91959 C1O0HF 71459392 IC50 = 43300 nM T91959 C31MUQ 71654770 IC50 > 50000 nM T91959 CU31DP 71654771 IC50 = 3.2 nM T91959 CAM70V 71654772 IC50 = 13 nM T91959 CE73FM 71654773 IC50 = 7.6 nM T91959 COV26M 71654774 IC50 = 56 nM T91959 CQ1KA4 71654775 IC50 = 8600 nM T91959 CMR87Y 71654838 IC50 > 50000 nM T91959 CAD5K9 71654839 IC50 = 4400 nM T91959 CTF4Y0 71654840 IC50 = 770 nM T91959 CU46KD 71654841 IC50 = 39 nM T91959 C4RA6P 71654842 IC50 = 280 nM T91959 C3WYU5 71654843 IC50 = 650 nM T91959 C12RAH 71654909 IC50 = 67 nM T91959 COW48U 71654910 IC50 = 92 nM T91959 C4AP1G 71654911 IC50 = 370 nM T91959 C1O0ZQ 71654912 IC50 = 61 nM T91959 CC6AJ7 71654913 IC50 = 28 nM T91959 CUHV94 71654914 IC50 = 30 nM T91959 CA2EM4 71654987 IC50 = 1300 nM T91959 CNU2D1 71654988 IC50 = 110 nM T91959 CU5HD4 71654989 IC50 = 2100 nM T91959 CP71AF 71654990 IC50 = 150 nM T91959 CUE91W 71654991 IC50 > 50000 nM T91959 CQOW51 71654992 IC50 > 50000 nM T91959 CS0FQ4 71654993 IC50 > 50000 nM T91959 CLDB05 71655060 IC50 = 4.9 nM T91959 C6JCD7 71655061 IC50 = 24 nM T91959 CX85ID 71655062 IC50 = 23 nM T91959 C8TX2W 71655063 IC50 = 29 nM T91959 C1TC4J 71655141 IC50 = 300 nM T91959 C6EFG7 73291970 IC50 = 3890 nM T91959 CMS0F6 73292335 IC50 = 8350 nM T91959 CMY90N 73292338 IC50 = 29400 nM T91959 CRZ62F 73355036 IC50 > 200000 nM T91959 C87LDV 77461130 IC50 > 100000 nM T91959 C67MJT 77461131 IC50 > 100000 nM T91959 C9YIS4 90654860 IC50 = 6000 nM T91959 C76QJZ 90654861 IC50 > 200000 nM T91959 CAD9C4 90654862 IC50 > 200000 nM T91959 C9U5QY 90654863 IC50 = 122000 nM T91959 CG6Z9E 90654864 IC50 > 200000 nM T91959 C5US4A 91673681 IC50 = 42200 nM T91959 CQO1F3 91673682 IC50 > 50000 nM T91959 CP43XT 101884802 IC50 = 33500 nM T91959 CSDE45 101884803 IC50 = 19300 nM T91959 CW3TR5 101884804 IC50 = 18300 nM T91959 C48DRM 101884805 IC50 = 22900 nM T91959 CKR05E 101884807 IC50 = 10400 nM T91959 CM40UV 101884808 Ki = 45 nM T91959 CA15KO 101884809 IC50 = 4370 nM T91959 CBJ50G 101884810 IC50 = 30100 nM T91959 CA7MT5 101884812 IC50 = 232000 nM T91959 C0W1CO 101884813 IC50 = 12300 nM T91959 CH06TS 101884814 IC50 = 2140 nM T91959 C2QJB4 101884815 IC50 = 16600 nM T91959 CZ17MX 101884816 IC50 = 9000 nM T91959 C2VX8K 112499922 IC50 > 100000 nM T91959 CL3X7K 118717122 IC50 = 27900 nM T91959 CY05KA 118717208 IC50 = 32500 nM T91959 CZQB67 118717209 IC50 = 33600 nM T91959 CCLI64 118722847 IC50 > 100000 nM T91959 CQM08D 121231415 IC50 = 1870 nM T91959 C0D2KV 121313586 IC50 = 177400 nM T91959 CVM95G 122186869 IC50 = 980 nM T91959 C5ZYP0 122186870 IC50 = 480 nM T91959 C97VZS 122186871 IC50 = 1100 nM T91959 CP5R3G 122186872 IC50 = 1400 nM T91959 CEOS03 122186873 IC50 = 320 nM T91959 C95ZQN 122186874 IC50 = 2100 nM T91959 CLO15R 122186875 IC50 = 3200 nM T91959 CML8G1 122186876 IC50 = 1910 nM T91959 C41TOB 122186877 IC50 = 1800 nM T91959 C57FWN 122186878 IC50 = 1620 nM T91959 CESR15 122186879 IC50 = 1750 nM T91959 C02XHR 122187733 IC50 = 1000 nM T91959 C5MGT9 122187734 IC50 = 450 nM T91959 C5XE4R 122187735 IC50 = 2100 nM T91959 CNIL28 122187736 IC50 = 890 nM T91959 C9KT4V 122187737 IC50 = 1440 nM T91959 CBAG46 122187738 IC50 = 800 nM T91959 CSU7W2 122187739 IC50 = 1290 nM T91959 C9J3MI 122187740 IC50 = 480 nM T91959 C2NEW8 122187741 IC50 = 360 nM T91959 CVX6G1 124155856 IC50 = 11500 nM T91959 C8R1KL 124155864 IC50 = 3330 nM T91959 CKU31X 124155865 IC50 = 2700 nM T91959 C1VNS9 124155880 IC50 = 2940 nM T91959 CI5SG4 124155887 IC50 > 200000 nM T91959 C8D6VI 124155892 IC50 = 15500 nM T91959 CE9HV7 124155894 IC50 = 3500 nM T91959 CL43GB 124155906 IC50 = 7120 nM T91959 C98FJW 124155909 IC50 = 1390 nM T91959 CG4KQ0 124155918 IC50 = 776 nM T91959 C2SK7Z 124155921 IC50 = 1220 nM T91959 CI3K8Z 124155944 IC50 = 6860 nM T91959 CC6E5F 124155947 IC50 = 3290 nM T91959 CDK5F1 124156051 IC50 = 2570 nM T91959 C5H1WI 124156054 IC50 = 6030 nM T91959 CK10FP 124156076 IC50 = 6390 nM T91959 CZ1X0F 124156082 IC50 = 8900 nM T91959 CN6YV0 124156084 IC50 = 843 nM T91959 C6VX3U 124156175 IC50 = 827 nM T91959 CA47GR 124156294 IC50 = 7510 nM T91959 C94NWB 124156297 IC50 = 5840 nM T91959 CLU7F3 124156311 IC50 > 200000 nM T91959 C25ACW 124156314 IC50 = 910 nM T91959 CC3H9B 124156319 IC50 = 5590 nM T91959 C0F8RC 124156322 IC50 = 723 nM T91959 CH2BJ7 124156324 IC50 = 2400 nM T91959 CC1B5Q 124156332 IC50 = 17700 nM T91959 CZ43QA 124156333 IC50 = 2500 nM T91959 CWT8L7 124156337 IC50 = 2710 nM T91959 C2CIJ9 124156338 IC50 = 28400 nM T91959 CU51OV 124156339 IC50 = 22300 nM T91959 CM64KZ 124156375 IC50 = 5620 nM T91959 CS8D4J 124156389 IC50 > 200000 nM T91959 CO71HP 124156406 IC50 = 4890 nM T91959 CTF86E 124156432 IC50 = 3390 nM T91959 CH2MQ3 124156454 IC50 = 8150 nM T91959 C5A1MN 124156461 IC50 = 9040 nM T91959 C4DR7M 124156464 IC50 = 829 nM T91959 C6Z3EX 124156466 IC50 = 9060 nM T91959 CQ1D7V 124156477 IC50 = 5580 nM T91959 CVG8H3 124156515 IC50 = 1770 nM T91959 CB6WM9 124156519 IC50 = 1560 nM T91959 C5X2EL 124156548 IC50 = 9660 nM T91959 COW18T 124156563 IC50 = 1590 nM T91959 C3R8OJ 124156568 IC50 = 5850 nM T91959 CJ2F5B 124156573 IC50 = 8240 nM T91959 CJ4C0I 124156580 IC50 = 106000 nM T91959 CF06XJ 124156582 IC50 = 7860 nM T91959 CJQC71 124156591 IC50 = 1080 nM T91959 C47GML 124156596 IC50 = 4110 nM T91959 CUJ71O 124156601 IC50 = 697 nM T91959 CK74XR 124156666 IC50 = 11400 nM T91959 CD83AZ 124156671 IC50 = 1620 nM T91959 COD08A 124156677 IC50 = 36200 nM T91959 C0R9GV 124156702 IC50 = 4080 nM T91959 CNT71Z 124156707 IC50 = 1880 nM T91959 C7I1AZ 124156715 IC50 = 18500 nM T91959 CZDJ49 124156728 Ki = 3400 nM T91959 CE1J6Y 124156731 IC50 = 503 nM T91959 COTD57 124156742 IC50 = 1560 nM T91959 CLA01I 124156756 IC50 > 200000 nM T91959 CP36XI 124156875 IC50 = 2370 nM T91959 C9KP4E 124156885 IC50 = 7320 nM T91959 CSM9Q8 124156886 IC50 = 6500 nM T91959 C2CI9E 124156887 IC50 = 1810 nM T91959 CUBJ73 124156888 IC50 = 5020 nM T91959 CV1R2F 124156892 IC50 = 3200 nM T91959 CULA86 124156896 IC50 = 85800 nM T91959 CFN1X9 124156913 IC50 = 7350 nM T91959 CH9R8A 124156914 IC50 = 8190 nM T91959 C4AXU0 124156920 IC50 = 17900 nM T91959 C4Y8GT 124156967 IC50 = 4790 nM T91959 C2DKH0 124157048 IC50 = 19500 nM T91959 C4G2NW 124157054 IC50 = 66400 nM T91959 CDR98I 124162056 IC50 = 4180 nM T91959 CU4IC8 126843233 IC50 > 100000 nM T91959 CU02IS 127027826 IC50 > 200000 nM T91959 CX9S6O 127032844 IC50 = 480 nM T91959 C8CV4N 127033814 IC50 = 269.5 nM T91959 C4J8WR 127034092 IC50 = 57.2 nM T91959 CH02OR 127034093 IC50 = 102.6 nM T91959 CJO78L 127034094 IC50 = 52.5 nM T91959 CY8TS5 127034095 IC50 = 42.9 nM T91959 C6FGW5 127034098 IC50 = 82.9 nM T91959 CCEP75 127034360 IC50 = 71 nM T91959 C84XPC 127048873 IC50 = 580 nM T91959 CBJD15 127049868 IC50 = 2640 nM T91959 C7P8JZ 129883511 IC50 > 50000 nM T91959 CZ45LV 129906245 IC50 > 50000 nM T91959 CCH2T8 129906312 IC50 = 9800 nM T91959 CY8B2P 132837649 IC50 = 10020 nM T91959 CA3L0T 134130520 IC50 > 1000000 nM T91959 CWV34S 134130814 IC50 = 470 nM T91959 C53GIN 134131007 IC50 = 54200 nM T91959 C8WD3G 134132512 IC50 = 3390 nM T91959 C2RX4P 134132760 IC50 = 2510 nM T91959 C7P4OF 134141051 IC50 = 3500 nM T91959 CYAK84 134141382 IC50 = 3820 nM T91959 C7B5KW 134142322 IC50 = 1820 nM T91959 CC4Z9Q 134143263 IC50 = 10800 nM T91959 CPKD12 134145576 IC50 = 1940 nM T91959 CN15TH 134148556 IC50 = 1480 nM T91959 CDBF51 134148882 IC50 = 56900 nM T91959 C53ATF 134148970 IC50 = 10000 nM T91959 CRON29 134150759 IC50 = 3180 nM T91959 C8MGQ9 134153152 IC50 = 3200 nM T91959 CZ8KH9 134155806 IC50 = 1060 nM T91959 CO2I4C 134433618 IC50 > 300000 nM T91959 C9YPF1 134820907 IC50 > 100000 nM T91959 CZR65A 135397670 IC50 > 100000 nM T91959 C64DLE 135397680 IC50 > 100000 nM T91959 CE3VW5 135659046 IC50 = 16700 nM T91959 CK5XC6 136240941 EC50 = 28600 nM T91959 C8YK2Z 137642096 IC50 = 17990 nM T91959 C9FN7L 137649628 IC50 = 11190 nM T91959 CLW0B7 137661474 IC50 > 100000 nM T91959 CAQ62X 137701235 Ki > 10000 nM T91959 CN2UH1 139303146 IC50 > 20000 nM T91959 CW7HG8 145960911 IC50 > 500000 nM T91959 CC0VT3 145962411 IC50 > 50000 nM T91959 CCXR94 145963449 IC50 = 4500 nM T91959 C5QIN6 145963700 IC50 > 500000 nM T91959 CX3MQ7 145965297 IC50 = 27910 nM T91959 C9XT0U 145966202 IC50 > 50000 nM T91959 C6W3YP 145966373 IC50 = 27030 nM T91959 CHQ8Z0 145967555 IC50 > 50000 nM T91959 C7ML9P 145967841 IC50 > 100000 nM T91959 CC3G2E 145970505 IC50 > 50000 nM T91959 C9CJ3Y 145971573 IC50 = 29240 nM T91959 CP1I5W 145972149 IC50 > 50000 nM T91959 CLT69F 145975278 IC50 = 23260 nM T91959 CWD0A9 145983712 Ki > 10000 nM T91959 C56MWZ 145986208 Ki > 10000 nM T91959 C8AS1P 155512143 IC50 > 100000 nM T91959 C80DBU 155512388 IC50 > 200000 nM T91959 CPZ01A 155512728 IC50 = 51000 nM T91959 CPQ48B 155513088 IC50 = 4200 nM T91959 CM6VN5 155513154 IC50 = 130 nM T91959 CZE29G 155514745 IC50 = 1600 nM T91959 C7VC1F 155517856 IC50 > 2000 nM T91959 CU0M1P 155518467 IC50 = 55 nM T91959 CN78HI 155519887 IC50 = 77 nM T91959 C2M5UT 155520367 IC50 = 770 nM T91959 C09RAW 155520570 IC50 = 1500 nM T91959 CFH1D8 155524740 IC50 > 100000 nM T91959 C4HV9G 155525499 IC50 = 110 nM T91959 C7H6XU 155528914 IC50 = 180 nM T91959 CTH59X 155529937 IC50 > 200000 nM T91959 CX8SC4 155530876 IC50 > 2000 nM T91959 C1JKR4 155531258 IC50 = 69200 nM T91959 C9WNP0 155531613 IC50 > 100000 nM T91959 CH30TZ 155546485 IC50 > 100000 nM T91959 C3WAN0 155550829 IC50 = 20.5 ug.mL-1 T91959 C2FZ1M 155550843 IC50 > 100000 nM T91959 C3D7GP 155554414 IC50 = 83000 nM T91959 C6FV9S 155554968 IC50 = 68000 nM T91959 C7IWD4 155564228 IC50 > 100000 nM T91959 C4CIL9 155564382 IC50 > 2000 nM T91959 D0E1QP 4262314 IC50 > 100000 nM T91959 D0E3NT 2130404 IC50 > 50000 nM T91959 D0M5FF 5083 IC50 = 3700 nM T24982 D02FEV 153965 IC50 = 2550 nM T24982 D02JIN 9823277 IC50 = 48 nM T24982 D09JXH 9831642 IC50 = 890 nM T24982 D0X8CH 53492727 IC50 = 42 nM T24982 CR0MV6 9810372 IC50 = 4 nM T24982 CJ7Q5F 9824764 IC50 = 3500 nM T24982 C3NIW1 9831643 IC50 = 0.28 nM T24982 C0GU5E 9852696 IC50 = 0.75 nM T24982 CY4M2Z 9865846 IC50 = 120 nM T24982 C0W9KT 9866565 IC50 = 5 nM T24982 CAR39S 9868843 IC50 = 7.3 nM T24982 C2J4LN 9887438 IC50 = 260 nM T24982 CFKC18 9894382 IC50 = 23 nM T24982 C3G2VH 9896647 IC50 = 2 nM T24982 CL65WP 9917720 IC50 = 2.3 nM T24982 CD4B3Y 9918280 IC50 = 1 nM T24982 C6CAM5 9934571 IC50 = 7 nM T24982 C4RQ6O 9936420 IC50 = 27 nM T24982 CW4MQ0 9938633 IC50 = 16 nM T24982 C0L8HG 9955824 IC50 = 2 nM T24982 CZ50NR 9961661 IC50 = 2 nM T24982 C52ZIB 9962161 IC50 = 1.6 nM T24982 CD76HT 10115455 IC50 = 2.2 nM T24982 CZC2K3 10168942 IC50 = 4 nM T24982 C1AH0C 10234233 IC50 = 770 nM T24982 C28ECJ 10280271 IC50 = 52 nM T24982 CX25KQ 10395459 IC50 = 1070 nM T24982 CYMF76 10479798 IC50 = 4400 nM T24982 CO68KA 11239135 IC50 = 1 nM T24982 CROW21 11495810 IC50 = 19 nM T24982 C9B7IL 11503193 IC50 = 8 nM T24982 CG0J9B 11505722 IC50 = 0.5 nM T24982 CZ2DA9 11505821 IC50 = 6 nM T24982 CDU3N5 11513254 IC50 = 8.5 nM T24982 CR7BN3 11517917 IC50 = 7.5 nM T24982 CKE58D 11518284 IC50 = 10 nM T24982 C82XEC 11519009 IC50 = 2 nM T24982 CEW3N0 11520475 IC50 = 2 nM T24982 C9E7JD 11532729 IC50 = 180 nM T24982 CHO08W 11533437 IC50 = 41 nM T24982 CHP7N4 11533566 IC50 = 17 nM T24982 CWB5P2 11535326 IC50 = 3 nM T24982 CI6G7Q 11538009 IC50 = 2000 nM T24982 C8O9VJ 11539289 IC50 = 46 nM T24982 C0HO7G 11539526 IC50 = 120 nM T24982 C47NUB 11540646 IC50 = 20 nM T24982 C9DA7V 11541489 IC50 = 0.3 nM T24982 C6AVN0 11541578 IC50 = 210 nM T24982 CGX0C7 11547864 IC50 = 7 nM T24982 C1R2AY 11548260 IC50 = 340 nM T24982 COX25D 11551679 IC50 > 50000 nM T24982 CKG56X 11561931 IC50 = 11 nM T24982 C73GCQ 11562188 IC50 = 320 nM T24982 C16NGA 11570280 IC50 = 28 nM T24982 CCP59O 11571157 IC50 = 18000 nM T24982 C0L9MV 11576438 IC50 = 1670 nM T24982 CTP93F 11577642 IC50 = 83 nM T24982 CG8D3F 11581857 IC50 = 90 nM T24982 C7Y6LE 11582766 IC50 = 90 nM T24982 CQJV49 11582797 IC50 = 190 nM T24982 CDX1M0 11583088 IC50 = 13 nM T24982 C34XHG 11583698 IC50 = 11 nM T24982 C60NUO 11588526 IC50 = 4000 nM T24982 CZS9C8 11595883 IC50 = 280 nM T24982 C16VQJ 11613677 IC50 = 600 nM T24982 CN06HE 11614719 IC50 = 4 nM T24982 C56TJZ 11618302 IC50 = 55 nM T24982 C16GOV 11620072 IC50 = 1300 nM T24982 CJY86Q 11620355 IC50 = 2670 nM T24982 C1R3CM 11621021 IC50 = 550 nM T24982 C2Y0WC 11621030 IC50 = 45 nM T24982 C7L3UD 11633742 IC50 = 50 nM T24982 C7BA2F 11635422 IC50 = 8.5 nM T24982 C81HAY 11639352 IC50 = 4800 nM T24982 CQ4HS9 11640949 IC50 = 5 nM T24982 C3O5VL 11641488 IC50 = 180 nM T24982 C5OP9X 11641507 IC50 = 22 nM T24982 C7O5KQ 11642769 IC50 = 220 nM T24982 CSI8D4 11646745 IC50 = 230 nM T24982 CFM5T2 11647331 IC50 = 54 nM T24982 C9OGT6 11648389 IC50 = 600 nM T24982 CZ5QE0 11648869 IC50 = 3.6 nM T24982 C7MVY6 11649102 IC50 = 1900 nM T24982 CXYE17 11663703 IC50 = 930 nM T24982 C4QVA8 11668567 IC50 = 21 nM T24982 CL6K8S 11670070 IC50 = 4.5 nM T24982 C2K4DS 11670901 IC50 = 75 nM T24982 CYI28E 11683733 IC50 = 5 nM T24982 C5U7ME 11686110 IC50 = 21000 nM T24982 CBKW96 11693232 IC50 = 9 nM T24982 CKW42F 11697828 IC50 = 180 nM T24982 CJU0R5 11698094 IC50 = 30 nM T24982 C6LF5B 11700336 IC50 = 260 nM T24982 C2GI9A 11705593 IC50 = 9.5 nM T24982 CSFI85 11705778 IC50 = 300 nM T24982 CO83MS 11705844 IC50 = 42 nM T24982 CDX91M 11705916 IC50 = 620 nM T24982 C5CRZ1 11706010 IC50 = 1000 nM T24982 C80FCD 11706316 IC50 = 400 nM T24982 C80KVB 11707494 IC50 = 4 nM T24982 CK3LJ9 11712315 IC50 = 318 nM T24982 C4TDA5 11721581 IC50 = 30 nM T24982 C3P8BY 20728332 IC50 = 70 nM T24982 CE35SL 23628193 IC50 = 2800 nM T24982 CB46QS 44326748 IC50 = 10800 nM T24982 C2JZM1 44326896 IC50 = 13300 nM T24982 CN0QV1 44326944 IC50 = 49000 nM T24982 C1OGH3 44327161 IC50 = 7100 nM T24982 C24JTI 44327162 IC50 = 9200 nM T24982 CRVQ83 44347821 IC50 = 1200 nM T24982 CK7PF6 44347832 IC50 = 1200 nM T24982 CMY94F 44347899 IC50 > 1000 nM T24982 CB2QU8 44347914 IC50 = 2500 nM T24982 CRUL41 44347940 IC50 = 310 nM T24982 CJ7P8Q 44347970 IC50 = 83 nM T24982 CEMJ37 44347971 IC50 = 320 nM T24982 C5PBO3 44348001 IC50 = 690 nM T24982 C6OY2Z 44348038 IC50 = 22 nM T24982 CTCW70 44348050 IC50 = 8 nM T24982 CO5C7X 44348051 IC50 = 26 nM T24982 CUQ4F2 44348052 IC50 = 6 nM T24982 C2F0RC 44348158 IC50 = 3 nM T24982 CGD26M 44348181 IC50 = 200 nM T24982 CL97QC 44348209 IC50 = 570 nM T24982 CBY60V 44348210 IC50 = 35 nM T24982 C18FUX 44348216 IC50 = 970 nM T24982 C8OF3Q 44348225 IC50 = 44 nM T24982 CTZV05 44348231 IC50 = 580 nM T24982 CM03AQ 44348386 IC50 = 320 nM T24982 CU7MI6 44392310 IC50 = 22000 nM T24982 CP8IA6 44392321 IC50 = 900 nM T24982 CW4K1S 44392322 IC50 = 1500 nM T24982 CI4CP8 44392323 IC50 > 300000 nM T24982 CU5W6D 44392324 IC50 > 300000 nM T24982 CJ42NL 44392345 IC50 > 300000 nM T24982 C45YDE 44392346 IC50 = 32000 nM T24982 CMT2Q5 44392360 IC50 = 60000 nM T24982 CK1J8G 44392368 IC50 = 1600 nM T24982 CIJ5C2 44392375 IC50 > 300000 nM T24982 CI6E8X 44403756 IC50 = 47 nM T24982 C75GPJ 44403760 IC50 = 8800 nM T24982 C75PRS 44403762 IC50 = 850 nM T24982 CZR2L0 44403764 IC50 = 7.5 nM T24982 CS2VH9 44403766 IC50 = 3.7 nM T24982 C5RC0H 44403793 IC50 = 16000 nM T24982 C2B1HR 44403803 IC50 = 59 nM T24982 CPR73S 44403804 IC50 = 68 nM T24982 C0IF5R 44404398 IC50 = 67 nM T24982 C50VKJ 45266101 IC50 = 2 nM T24982 CDB0K3 45266104 IC50 = 5.7 nM T24982 C2CZF4 45266105 IC50 = 3 nM T24982 C7L9CU 45266106 IC50 = 7 nM T24982 CG3D6V 45266107 IC50 = 5500 nM T24982 CR91GD 45266108 IC50 = 0.76 nM T24982 C71NQP 49799588 Ki = 1910 nM T24982 C1NWI9 49799589 Ki = 2020 nM T24982 C0A2QL 49799590 Ki = 2310 nM T24982 CYIA04 49799591 Ki = 1250 nM T24982 CP1T8A 49799592 Ki = 3020 nM T24982 CD56QV 49799593 Ki = 2630 nM T24982 CQ5ZP3 49799594 Ki = 889 nM T24982 CL5JV9 49799595 Ki = 3200 nM T24982 CT7B9L 49799596 Ki = 3890 nM T24982 C7E0VZ 49799597 Ki = 4220 nM T24982 C4GC3B 49799598 Ki = 6090 nM T24982 CMGK52 49799599 Ki = 3930 nM T24982 CQ6FJ2 49799600 Ki = 587 nM T24982 C1ALH5 49799601 Ki = 275 nM T24982 C1S9DJ 49799602 Ki = 2300 nM T24982 CX18KE 49799610 Ki = 7650 nM T24982 CJY4N5 49799611 Ki = 4030 nM T24982 CDYU58 49799616 Ki = 2640 nM T24982 C5K1HP 49799617 Ki = 16300 nM T24982 C4CVP7 49799618 Ki = 15900 nM T24982 C3FV2L 49799619 Ki = 3160 nM T24982 CK5F1G 49799620 Ki = 8070 nM T24982 CYO8F4 49799621 Ki = 4300 nM T24982 C6IGQ2 49799622 Ki = 5190 nM T24982 C1SO9B 49799624 Ki = 40400 nM T24982 CA6S0Y 49799625 Ki = 35900 nM T24982 CU2N8M 49799626 Ki = 108000 nM T24982 CP81TN 49799627 Ki = 126000 nM T24982 CA6F3P 49799628 Ki = 41000 nM T24982 CKS42G 56660067 Ki = 1150 nM T24982 CCJT38 56665024 Ki = 5160 nM T24982 C9CKO2 56667635 Ki = 2240 nM T24982 C9GD6O 56671164 Ki = 6530 nM T24982 C5J0QE 56677822 Ki = 5260 nM T24982 CP80IW 56681532 Ki = 2010 nM T24982 C0J8CX 67460562 IC50 = 17 nM T24982 CAI8Y9 67463812 IC50 > 3000 nM T24982 CHI50P 67463839 IC50 = 51 nM T24982 C36DQP 67464261 IC50 > 3000 nM T24982 CIE2C9 67464286 IC50 = 41 nM T24982 C96SWC 67464325 IC50 = 1458 nM T24982 CR1DT0 67464354 IC50 = 59 nM T24982 C47WQC 67464917 IC50 = 2698 nM T24982 C8AYV2 67465761 IC50 = 245 nM T24982 CA40PJ 67465799 IC50 = 51 nM T24982 C26KGC 67465816 IC50 = 97 nM T24982 CFK1I4 67465851 IC50 > 3000 nM T24982 C2JI0L 67465855 IC50 = 2 nM T24982 C6NLH1 67465879 IC50 = 425 nM T24982 CHU5G6 67465944 IC50 = 728 nM T24982 C2EG6F 67465957 IC50 = 1287 nM T24982 CR84EL 67465998 IC50 = 751 nM T24982 CXNG13 67466300 IC50 = 6 nM T24982 C2TO1A 67466465 IC50 > 3000 nM T24982 CNW9I4 67466860 IC50 = 2540 nM T24982 CMI0X2 68207767 IC50 = 190 nM T24982 CAP79G 68207809 IC50 = 47 nM T24982 C1BW8A 68207860 IC50 > 3000 nM T24982 CL2D0Z 71237450 IC50 = 249 nM T24982 C5OPM6 71237501 IC50 = 276 nM T24982 CQB42P 71237567 IC50 = 23 nM T24982 CN2DQ9 71237740 IC50 = 55 nM T24982 CBJ6D4 71237989 IC50 = 32 nM T24982 CI2H6N 71238092 IC50 = 4 nM T24982 CIE71J 71238099 IC50 = 367 nM T24982 C2N5WV 71599441 IC50 > 25118.86 nM T24982 C58NVG 71660821 IC50 > 25118.86 nM T24982 C5I0NP 71733736 IC50 = 54 nM T24982 CF9X1B 71733926 IC50 = 365 nM T24982 CH7N8X 71733927 IC50 > 3000 nM T24982 CDZ3S6 71734215 IC50 = 4 nM T24982 C0JZD1 71734218 IC50 = 2 nM T24982 C1J9EK 71734311 IC50 = 167 nM T24982 C24NJQ 71734313 IC50 = 128 nM T24982 CO31ZU 71734502 IC50 = 34 nM T24982 C7MCZ8 71734588 IC50 = 13 nM T24982 CH9RV5 71734589 IC50 = 4 nM T24982 C9ZV7L 71734590 IC50 = 50 nM T24982 C21IOX 71734591 IC50 = 900 nM T24982 C96GPJ 71734592 IC50 = 44 nM T24982 CRJK43 71734683 IC50 = 133 nM T24982 CO37FH 71734684 IC50 = 4 nM T24982 CRJ69A 71734776 IC50 = 11 nM T24982 CMZ90C 71734851 IC50 = 9 nM T24982 C0DEA1 145974037 IC50 > 25118.86 nM T28925 D0F0ZE 153241 IC50 = 7 nM T28925 CUY74W 27513 IC50 = 99000 nM T28925 C3N8UF 70133 IC50 = 620000 nM T28925 CMB1D2 80063 IC50 = 31000 nM T28925 CG68LK 94711 IC50 = 168000 nM T28925 CD68XC 104251 IC50 = 54000 nM T28925 C8SH7I 188321 Ki = 62000 nM T28925 C8IOM3 230282 IC50 = 32000 nM T28925 CQ8I0A 3718102 IC50 = 21000 nM T28925 C75FLA 9797026 IC50 = 40 nM T28925 CKY2D7 9901690 IC50 = 180 nM T28925 C0AJ8G 11779435 IC50 = 32000 nM T28925 CFLV58 15625188 IC50 = 20 nM T28925 C94MKX 20766827 IC50 = 1300 nM T28925 CK50VP 20766837 IC50 = 2400 nM T28925 CIVN94 20766838 IC50 = 15000 nM T28925 CX30TQ 20766839 IC50 = 430 nM T28925 C7JW5O 20766920 IC50 = 8100 nM T28925 CG7R1S 20766923 IC50 = 35000 nM T28925 C0V5BJ 20766925 IC50 = 27000 nM T28925 CVR34M 20766928 IC50 = 14000 nM T28925 CIK04R 22558406 IC50 = 20000 nM T28925 C4LOX1 22558440 IC50 = 470 nM T28925 C05CKF 44291510 IC50 = 910 nM T28925 CH71MA 44291528 IC50 = 730 nM T28925 CQB23X 44291630 IC50 = 88000 nM T28925 CG0AS8 44291704 IC50 = 18000 nM T28925 C7C3KX 44291706 IC50 = 16000 nM T28925 CA5IS0 44291905 IC50 = 200 nM T28925 CYC57I 44291978 IC50 = 1200 nM T28925 C98QUE 44292362 IC50 = 4400 nM T28925 CVO9E5 44331477 IC50 = 7 nM T28925 C8O6NZ 135887992 Ki = 38000 nM T28925 C9E1TW 135976435 Ki = 1110 nM T28925 C2U5QN 135976440 Ki = 120000 nM T28925 CBOZ73 135976442 Ki = 190000 nM T28925 CG63EX 135976453 Ki = 46000 nM T28925 C25EPJ 135976460 Ki = 600000 nM T28925 D0H2YT 135398640 Ki = 250 nM T28925 D0L0ZP 15462732 IC50 = 19000 nM T28925 D0Z8EV 446541 IC50 = 20000 nM T04210 C3H5DF 7172 EC50 = 6600 nM T04210 CJUD30 7728970 EC50 = 37300 nM T04210 CJY35N 10102480 EC50 = 0.3388 nM T04210 CTE84B 10260704 EC50 = 0.71 nM T04210 CRF1I2 10351235 EC50 = 0.4 nM T04210 CK56IA 13920660 EC50 = 34.3 nM T04210 C39FCZ 13920665 IC50 = 802.9 nM T04210 CZM45J 13920666 EC50 = 616.1 nM T04210 CH82QU 13920670 EC50 = 2495 nM T04210 CO7X1P 45277088 Ki < 10000 nM T04210 C26EWX 45277089 Ki < 10000 nM T04210 C6X4ER 45277090 Ki < 10000 nM T04210 CH7I1J 45277245 Ki < 10000 nM T04210 C8FO0Q 87415277 EC50 = 0.2 nM T04210 C4LZ8G 87415284 EC50 = 0.37 nM T04210 CMFU53 88563444 EC50 = 0.82 nM T04210 C9K4XR 101879981 EC50 = 14000 nM T04210 C4QSN7 102340758 EC50 = 3.8 nM T04210 COA2W3 117072558 EC50 = 2.6 nM T04210 CAX3W4 118708073 EC50 = 8.4 nM T04210 CGH1K9 118708139 EC50 = 0.7943 nM T04210 CB8NX1 118716778 EC50 = 31100 nM T04210 CH7TK3 118716779 EC50 = 73000 nM T04210 CKI1S6 118716780 EC50 = 253000 nM T04210 CR5O7X 118716784 EC50 = 47000 nM T04210 CT7E1P 118721282 EC50 = 391 nM T04210 CFH73K 126558991 EC50 = 10.23 nM T04210 C4LTY5 127025171 EC50 = 281.84 nM T04210 C2Y8WJ 127025772 EC50 = 724.44 nM T04210 C4B7GF 127026380 EC50 = 107.15 nM T04210 CS7H6Y 127026692 EC50 = 2511.89 nM T04210 C39QJN 127026693 EC50 = 56.23 nM T04210 CS4M3H 127027325 EC50 = 10000 nM T04210 CDA87B 127028302 EC50 = 0.2138 nM T04210 C09HYQ 127029245 EC50 = 42.66 nM T04210 C7PDT0 137633449 EC50 = 0.22 nM T04210 CAYE32 137633990 EC50 = 9.3 nM T04210 C9J6MS 137634038 EC50 = 1.4 nM T04210 C4MP6D 137635007 EC50 = 0.34 nM T04210 CV0SA3 137635179 EC50 = 1.2 nM T04210 C9A1NV 137636126 EC50 = 3.4 nM T04210 CZ4ER6 137636135 EC50 = 1.8 nM T04210 CEZI98 137636174 EC50 = 0.8 nM T04210 C0V4QH 137636908 EC50 = 0.47 nM T04210 CI3EN9 137637194 EC50 = 0.31 nM T04210 CO5KI9 137638792 EC50 = 0.94 nM T04210 CI8Z6A 137639361 EC50 = 11 nM T04210 C60GTH 137639547 EC50 = 7.3 nM T04210 CZA43W 137640394 EC50 = 0.83 nM T04210 CH0M4E 137640682 EC50 = 0.41 nM T04210 C8EPD9 137640690 EC50 = 0.2 nM T04210 C3SY4E 137640722 EC50 = 3.5 nM T04210 C0BR5G 137642468 EC50 = 8.4 nM T04210 C1NZS2 137642598 EC50 = 4.1 nM T04210 CEZO84 137642989 EC50 = 0.28 nM T04210 C8Z5TV 137643044 EC50 = 0.58 nM T04210 C6D5PN 137643754 EC50 = 0.42 nM T04210 C62VJS 137643907 EC50 = 0.39 nM T04210 CZW4O1 137644441 EC50 = 3.3 nM T04210 C7LTU5 137645284 EC50 = 2 nM T04210 CB4PL6 137646480 EC50 = 12 nM T04210 CA91FH 137646678 EC50 = 0.16 nM T04210 CY9VN0 137647003 EC50 = 1.5 nM T04210 C9SRK0 137647843 EC50 = 3.8 nM T04210 CMZO51 137651400 EC50 = 9.4 nM T04210 C6BZ4Q 137652197 EC50 = 4.2 nM T04210 C4IZF9 137652435 EC50 = 0.43 nM T04210 C41GTA 137652696 EC50 = 0.69 nM T04210 C02CQP 137652739 EC50 = 0.93 nM T04210 CX1O2U 137654882 EC50 = 1.9 nM T04210 C2GCF6 137654963 EC50 = 6.2 nM T04210 C23CJO 137656685 EC50 = 5.8 nM T04210 CIOB49 137657622 EC50 = 3.6 nM T04210 CHVG89 137660286 EC50 = 0.74 nM T04210 C1PA4N 137660608 EC50 = 3 nM T04210 CC0DM7 137660871 EC50 = 0.15 nM T04210 C3U2AG 137662007 EC50 = 0.57 nM T04210 CXU43I 145948899 EC50 = 1.905 nM T04210 CGC6I4 145948939 EC50 = 6309.57 nM T04210 CJ90ZA 145948940 EC50 = 107.15 nM T04210 C1XUP6 145948945 EC50 = 6309.57 nM T04210 CXL19B 145948995 EC50 = 1000 nM T04210 C6T9KU 145949005 EC50 = 794.33 nM T04210 CI3CP8 145949312 IC50 = 13 nM T04210 CJE9N8 145949890 EC50 = 0.83 nM T04210 CMXF70 145950449 EC50 = 6.2 nM T04210 C08LUS 145950548 EC50 = 472.1 nM T04210 C7HT6J 145950907 IC50 = 598.9 nM T04210 CJX82E 145950926 IC50 = 1019 nM T04210 CH40RP 145951399 EC50 = 382.3 nM T04210 CH9E5Y 145951684 EC50 = 13.4 nM T04210 CE0H7Z 145952282 EC50 = 59.7 nM T04210 C5JNT2 145952841 EC50 = 250 nM T04210 C13JWO 145953216 IC50 = 1813 nM T04210 CN17CJ 145953723 EC50 = 1.8 nM T04210 C1VAK6 145953783 EC50 = 5.4 nM T04210 CYXG32 145954208 EC50 = 1993 nM T04210 C0PZ9I 145954222 EC50 = 3.5 nM T04210 CJ9IZ8 145954330 EC50 = 1286 nM T04210 C5WO9C 145955290 EC50 = 192.6 nM T04210 CSZR24 145955540 EC50 = 624.3 nM T04210 CMVI71 145956001 EC50 = 1103 nM T04210 CJ1FS2 145956177 IC50 = 29.1 nM T04210 C5C9QN 145956751 EC50 = 1.6 nM T04210 C4EKH3 145957679 EC50 = 1407 nM T04210 C3LE8D 145958000 EC50 = 459.3 nM T04210 C80IPJ 145958151 EC50 = 225.7 nM T04210 C0YGX7 145958189 EC50 = 55.6 nM T04210 CN9M8W 145958420 IC50 = 1365 nM T04210 C7R5OF 145958560 IC50 = 1089 nM T04210 CS3DU2 145958712 EC50 = 3.8 nM T04210 CQ23YK 145959083 EC50 = 382.2 nM T04210 C8KW6U 145959164 EC50 = 1830 nM T04210 C3P6KU 145959336 IC50 = 465.5 nM T04210 CPS2V1 145959590 IC50 = 28.8 nM T04210 CM8EN5 145959730 EC50 = 339.2 nM T04210 CC6I9T 145959831 IC50 = 1857 nM T04210 C0XDK3 145959870 EC50 = 28.6 nM T04210 COJ4G1 145960270 EC50 = 4.8 nM T04210 CZYI89 145960563 IC50 = 39.1 nM T04210 C48HCB 145971434 IC50 = 195.3 nM T04210 C3F4IC 145971940 EC50 = 926.3 nM T04210 CEFK04 145972185 EC50 = 378 nM T04210 CX6Q5M 145972641 EC50 = 440.8 nM T04210 CXS39Z 145972936 EC50 = 0.7 nM T04210 CQ3M5K 145973626 EC50 = 10.2 nM T04210 C9IJP3 145974070 IC50 = 261.6 nM T04210 C12QJH 145974338 EC50 = 242.2 nM T04210 D09ALJ 5280805 EC50 = 1200 nM T27944 D0V2GT 5311023 Ki > 5000 nM T27944 C9NG4X 16033 EC50 = 0.03 nM T27944 C74KDN 624746 IC50 > 10000 nM T27944 C39UDN 5312114 IC50 = 5740 nM T27944 CI26VT 9799669 IC50 > 30000 nM T27944 C5MC8Y 9802119 IC50 > 10000 nM T27944 CK7QY8 9867212 IC50 > 30000 nM T27944 C0EGK5 9869458 Ki > 5000 nM T27944 CPGD84 9887225 IC50 > 10000 nM T27944 CS92LR 9916525 Ki > 10000 nM T27944 CH1Q6E 10008757 Ki > 10000 nM T27944 CK3W5X 10030299 Ki > 10000 nM T27944 C73QBA 10047509 IC50 > 10000 nM T27944 CL96TH 10110741 IC50 > 10000 nM T27944 C6IXU4 10293988 Ki > 10000 nM T27944 C8L7WY 10295464 IC50 > 30000 nM T27944 CA1C6E 10418848 Ki = 5.8 nM T27944 C84MSG 10524003 Ki > 10000 nM T27944 CKQ2G1 10531484 Ki > 10000 nM T27944 CQ1P5I 10554658 Ki > 10000 nM T27944 C0F9SD 10555187 Ki > 10000 nM T27944 C0FP2G 10619067 Ki > 10000 nM T27944 CZ0U1P 10625004 Ki > 10000 nM T27944 C3L6TA 10671331 Ki > 10000 nM T27944 C7MC2O 10672357 Ki > 10000 nM T27944 C6HQ1X 10692519 Ki > 10000 nM T27944 CS4JF0 10820168 Ki = 3737 nM T27944 CEH6O1 10820196 Ki = 2403 nM T27944 CQ49SB 11640844 Ki > 10000 nM T27944 CJ5TE0 11798404 Ki > 10000 nM T27944 CUM43R 12071667 IC50 > 10000 nM T27944 CIYU59 20587808 IC50 > 10000 nM T27944 CEOA23 22254020 IC50 > 1000 nM T27944 CBS20U 22254050 IC50 > 1000 nM T27944 CO32YX 22254068 IC50 > 1000 nM T27944 CHQT84 22254131 IC50 > 1000 nM T27944 CP7E2N 22325336 IC50 > 10000 nM T27944 CBS23H 24868176 Ki = 0.37 nM T27944 CG3VL7 25067562 IC50 > 10000 nM T27944 C7IH3J 25181112 Ki > 10000 nM T27944 C7VID1 25211875 IC50 > 10000 nM T27944 CNU7P4 42630820 IC50 > 10000 nM T27944 CJM96N 44461116 IC50 > 30000 nM T27944 C68NXC 44517723 IC50 > 10000 nM T27944 CZ65XF 44579887 IC50 > 10000 nM T27944 CVO10S 44580050 IC50 > 10000 nM T27944 C30LDO 45487447 IC50 > 10000 nM T27944 CL9PW1 45487448 IC50 > 10000 nM T27944 C5YB1P 46231125 Ki = 5.8 nM T27944 CZD7T5 46880224 Ki > 10000 nM T27944 CH5A3Z 52953217 Ki > 3000 nM T27944 CV10HR 52953219 Ki > 500 nM T27944 C97QRD 54582344 Ki > 5000 nM T27944 CLQ9Y2 56841989 Ki = 0.79 nM T27944 C8QO1W 71719108 Ki > 7500 nM T27944 C9UH7J 72205287 Ki > 5000 nM T27944 CL8NG4 72205482 Ki > 5000 nM T27944 CDZU03 72205484 Ki > 5000 nM T27944 CH2VP3 72205486 Ki = 3800 nM T27944 CAK56G 72205667 Ki > 5000 nM T27944 CB57PL 72205867 Ki = 150 nM T27944 CFC0Q6 72206048 Ki > 5000 nM T27944 CFV1X0 72711815 EC50 = 451 nM T27944 CE6KV1 72712030 EC50 = 94 nM T27944 C1X2AR 73346549 Ki > 5000 nM T27944 C3Y8HL 73349568 Ki > 5000 nM T27944 CPXJ28 73349570 Ki = 3200 nM T27944 C0NM1P 73351119 EC50 = 291 nM T27944 CM5ZV2 73351127 Ki > 5000 nM T27944 C7TL4C 73352596 Ki > 5000 nM T27944 C27BRN 73352597 Ki = 2000 nM T27944 CRC73X 73354075 Ki = 50 nM T27944 CRL10F 73354088 Ki = 3700 nM T27944 CL5A3F 73354090 Ki > 5000 nM T27944 CIFL82 73354092 Ki = 3300 nM T27944 C9XCU8 73354094 Ki = 3500 nM T27944 CCK72G 73355613 Ki = 4100 nM T27944 C4FDT1 73355615 Ki > 5000 nM T27944 CO26NJ 73355617 Ki = 390 nM T27944 CUM6D5 73357147 Ki = 35 nM T27944 CXJ85A 73357158 Ki > 5000 nM T27944 CB3FG4 85472343 Ki = 2.3 nM T27944 CW2BG8 127029975 Ki = 3.5 nM T27944 C0HX5P 127030358 Ki = 3.6 nM T27944 C7Q2WP 127030359 Ki = 0.66 nM T27944 COJD62 127031280 Ki = 1.5 nM T27944 CK0A1M 127031281 Ki = 1.2 nM T27944 CYO6S0 127032107 Ki = 7.4 nM T27944 C0XR6M 127041306 Ki > 10000 nM T27944 C5PA2G 127041908 Ki > 10000 nM T27944 C7TM1Y 127042243 Ki > 10000 nM T27944 C62JIE 127042244 Ki > 10000 nM T27944 C9L6CZ 131886627 Ki = 1.06 nM T27944 C9WG7C 145948675 Ki = 0.5 nM T27944 C8ZAN2 145979152 Ki = 0.1 nM T27944 C4SB9P 145979291 Ki = 630 nM T27944 CQ78WY 145979469 Ki = 1000 nM T27944 CO1M3D 145979616 Ki = 2500 nM T27944 C3OXL9 145979975 Ki = 199.53 nM T27944 C4H9BZ 145980763 Ki = 15.85 nM T27944 CH5MZ8 145980782 Ki = 630 nM T27944 CI5F7E 145980802 Ki = 630 nM T27944 CP4RI5 145980997 Ki = 0.1585 nM T27944 CW80EN 145981168 Ki = 5000 nM T27944 CTF1C6 145981319 Ki = 6.3 nM T27944 COB75I 145981742 Ki = 25 nM T27944 C60AUT 145981829 EC50 > 1000 nM T27944 COF9U8 145982156 Ki = 2500 nM T27944 CXE2K1 145984150 Ki = 790 nM T27944 CM4VG2 145984378 Ki = 316.23 nM T27944 CG74XB 145985156 Ki = 63 nM T27944 C5XL9U 145985176 Ki = 0.01 nM T27944 C63DRI 145985639 Ki = 1584.89 nM T27944 C5UDH2 145986414 Ki = 316.23 nM T27944 CLEQ40 145986472 Ki = 12.59 nM T27944 CZ68SU 145986539 Ki = 1584.89 nM T27944 CGB4Y3 145987289 Ki = 5000 nM T27944 CI1XY0 145987577 Ki = 100 nM T27944 C4T5IJ 145987618 Ki = 2500 nM T27944 CL2I3Y 145987802 Ki = 500 nM T27944 CIZ94Y 145988210 Ki = 0.1585 nM T27944 CRW15D 145989250 Ki = 50 nM T27944 C5O8AZ 145989327 Ki = 790 nM T27944 CG63IW 145989789 Ki = 1995.26 nM T27944 CF5OV2 145990257 EC50 > 1000 nM T27944 CH50MF 145991293 EC50 > 1000 nM T27944 CDX86E 145991438 Ki = 1258.93 nM T27944 C6PS8F 145991876 Ki = 1000 nM T27944 C7K8CT 145992181 Ki = 2.5 nM T27944 CC72HP 145992661 Ki = 0.01 nM T27944 C5KF0O 145992989 Ki = 125.89 nM T27944 CQH29C 145993358 Ki = 1.585 nM T27944 C9Z4PM 145993376 Ki = 125.89 nM T27944 CAZ6I7 145993698 Ki = 100 nM T27944 CPD7M9 145994220 Ki = 50 nM T27944 C4AB9K 155512045 IC50 = 616.6 nM T27944 CP9OE1 155513842 EC50 = 33.11 nM T27944 CHW62U 155517347 EC50 = 30.2 nM T27944 C4KN0H 155517812 EC50 = 5.129 nM T27944 C71AMJ 155521784 Ki = 32.36 nM T27944 C2BUO8 155523949 EC50 = 6.761 nM T27944 CQF01J 155524657 Ki = 0.18 nM T27944 C35VJX 155525593 IC50 = 2.291 nM T27944 CGHC94 155532134 IC50 = 93.33 nM T27944 CY8MK6 155533017 EC50 = 23.44 nM T27944 C3AF1H 155533076 Ki = 4.169 nM T27944 C2VJ4Y 155537755 EC50 = 12.88 nM T27944 C2GBO9 155541756 EC50 = 7.586 nM T27944 CCK32B 155543070 Ki = 0.32 nM T27944 C5FIG6 155543507 EC50 = 5.495 nM T27944 C5A7BF 155546907 EC50 = 30.2 nM T27944 CCZ09U 155547323 Ki = 11 nM T27944 C1T7DH 155549336 Ki = 2.8 nM T27944 CS8MB4 155553670 EC50 = 3.715 nM T27944 CDT81L 155553742 EC50 > 3000 nM T27944 C7Q6NB 155553966 EC50 = 95.5 nM T27944 CL5G9Y 155557501 IC50 = 70.79 nM T27944 CVI2M6 155557900 IC50 = 23.99 nM T27944 CX43VE 155561277 EC50 > 3000 nM T27944 C4M9NL 155561620 Ki = 12 nM T27944 C86FRY 155563387 EC50 = 37.15 nM T27944 CH4XA1 155564444 Ki = 912.01 nM T27944 CC8WB6 155565033 EC50 = 4.266 nM T27944 D00OLA 44409453 Ki = 3.9 nM T27944 D07OOG 73347134 Ki = 2 nM T27944 D08YWE 73348635 Ki = 4.1 nM T27944 D0G4HT 73354703 Ki = 0.05 nM T27944 D0J9VA 44409452 Ki = 5.3 nM T27944 D0U5TK 5311022 Ki > 5000 nM T27944 D0V0HM 73345612 Ki = 4.2 nM T26623 D03KOZ 1549120 IC50 = 0.03 ug.mL-1 T26623 D04AIT 5280445 IC50 = 600 nM T26623 D05FTJ 4044 IC50 = 77000 nM T26623 D07HBX 338 IC50 > 1000000 nM T26623 D08EBN 41684 IC50 = 8220 nM T26623 D09BHB 5509 IC50 = 2390 nM T26623 D0B2WJ 3371 IC50 = 41000 nM T26623 D0K8KX 5280343 IC50 = 1.05 ug.mL-1 T26623 D0R1RS 3715 IC50 = 6000 nM T26623 D0TG1H 3033 IC50 > 100000 nM T26623 D0W9WF 3825 IC50 = 180000 nM T26623 D0Z5IU 1548887 IC50 = 374 nM T26623 D00EWR 160024 IC50 = 9 nM T26623 D04BFU 157839 IC50 = 5 nM T26623 D04PBH 5280804 IC50 = 4500 nM T26623 D0K8TI 153948 IC50 = 15 nM T26623 D0L4FS 5280961 IC50 = 20000 nM T26623 D0Q7QY 53359 IC50 = 10 nM T26623 D0R9YR 64971 IC50 = 11000 nM T26623 D0T4SG 11292191 IC50 = 794 nM T26623 D0Z0HH 3503 Ki = 500 nM T26623 D0M9RE 6420118 IC50 = 0.84 nM T26623 D0N7BW 1276529 IC50 = 20.2 nM T26623 D02CGC 337359 IC50 = 120 nM T26623 D03PIB 2120 IC50 = 6500 nM T26623 D06EDT 1613 IC50 = 3.1 nM T26623 D0C7KK 5724 IC50 = 42.4 nM T26623 D0J6JZ 190816 IC50 = 12.2 nM T26623 D0Q7AW 65673 IC50 = 54.7 nM T26623 D0U7OU 3220 Ki = 2113 nM T26623 D0U9TM 5278 IC50 = 21 nM T26623 CI0WH9 72 IC50 = 42.7 ug.mL-1 T26623 CAY34Q 999 IC50 = 96000 nM T26623 CJK48W 5252 IC50 = 20000 nM T26623 CX45NQ 8892 IC50 = 68200 nM T26623 CQYO59 11970 IC50 = 3500 nM T26623 CL70CJ 13650 IC50 = 62000 nM T26623 CW5Z8A 41531 IC50 = 330 nM T26623 C7NG8I 43585 IC50 = 700 nM T26623 C97DVT 81058 IC50 = 4400 nM T26623 CF2L6T 92525 IC50 = 1.15 ug.mL-1 T26623 CA9YN2 99477 IC50 = 171000 nM T26623 CHF2E5 101761 IC50 = 84000 nM T26623 C2R4AE 114776 IC50 = 1910 nM T26623 C32DAX 119307 IC50 = 147300 nM T26623 CEYH47 122660 Ki = 7300 nM T26623 C7MCR1 124021 IC50 = 8000 nM T26623 CE2C6D 132323 IC50 = 5.2 nM T26623 C4IRY2 164676 IC50 = 8690 nM T26623 CO94ZR 164853 IC50 = 6900 nM T26623 C40GZU 173910 IC50 = 3100 nM T26623 CF6AY3 176053 IC50 = 22 nM T26623 CS61XQ 214654 IC50 = 4100 nM T26623 C7BRG3 259386 Ki = 56000 nM T26623 C8N5IM 293170 Ki = 48000 nM T26623 C0SMD7 339231 IC50 = 6400 nM T26623 CKYQ94 375713 Ki = 1500 nM T26623 CUF5O9 390735 IC50 >= 10000 nM T26623 C7HME8 439246 IC50 = 28870 nM T26623 CFJ58L 447950 IC50 = 72.6 nM T26623 CG24QH 449156 IC50 = 570 nM T26623 CYPW07 471004 IC50 > 194400 nM T26623 CZ0AH3 638278 IC50 = 320 nM T26623 C1Q3CE 685919 IC50 = 57 nM T26623 C1N0ZJ 1201064 IC50 = 0.13 nM T26623 CS2T8A 1201074 IC50 = 0.82 nM T26623 CCXP42 1201110 IC50 = 125 nM T26623 CXNA13 1201165 IC50 = 25 nM T26623 C0B3ZE 1201317 IC50 = 40 nM T26623 CH82ZT 1201321 IC50 = 53 nM T26623 CS7UW2 1206233 IC50 = 0.15 nM T26623 CFX90H 1243769 IC50 = 13280 nM T26623 C9XDJ0 1350369 IC50 = 279.9 nM T26623 C50QEB 1351632 IC50 = 0.49 nM T26623 CO7M2D 1351633 IC50 = 150 nM T26623 C6UZ1A 1383990 IC50 = 52 nM T26623 C30CVQ 1622257 IC50 = 78 nM T26623 CTHY21 2176938 IC50 = 0.26 nM T26623 C2FZ4N 2377118 IC50 = 10200 nM T26623 C45KNE 2403877 IC50 = 2760 nM T26623 C1X5DE 2415512 IC50 = 1950 nM T26623 C3F2IJ 2462392 IC50 = 1130 nM T26623 CGOQ53 2622535 IC50 = 720 nM T26623 CAKX74 4763851 IC50 > 50000 nM T26623 C4JQ5B 4763963 IC50 = 50000 nM T26623 CLZ13P 5280441 IC50 = 566660 nM T26623 CNZ73E 5280567 IC50 = 24500 nM T26623 CH50QK 5281643 IC50 = 3000 nM T26623 C57OTP 5281691 IC50 = 2700 nM T26623 CJLF09 5281702 IC50 = 2030 nM T26623 CGS9B0 5281780 IC50 = 78 nM T26623 CMAH08 5315472 IC50 = 5100 nM T26623 CFB0N1 5318591 IC50 = 720 nM T26623 CRY76T 5319502 IC50 = 64400 nM T26623 C5S4KV 5320203 IC50 = 66300 nM T26623 C1RUA2 5320844 IC50 = 95310 nM T26623 CFXB53 5338490 IC50 = 20800 nM T26623 C2SE9J 5369459 IC50 = 23000 nM T26623 C4T5NB 5376802 IC50 = 5000 nM T26623 CX0I3E 5393159 IC50 = 63300 nM T26623 CVFQ91 5479463 IC50 = 1800 nM T26623 CIC8S7 5490064 IC50 = 19050 nM T26623 CFV8Y1 5919576 IC50 = 400 nM T26623 C1ILT3 5933486 IC50 = 194 nM T26623 C0XGU4 6006931 IC50 = 6140 nM T26623 CU8T4O 6056260 IC50 = 8953.65 nM T26623 C6YG8U 6229410 IC50 = 480 nM T26623 CSG8D7 6440361 IC50 = 38000 nM T26623 CSA24L 6474310 IC50 = 88 nM T26623 C2M4FJ 9800756 IC50 = 7 nM T26623 CXS1G2 9804333 IC50 = 15 nM T26623 CGY1M4 9805341 IC50 = 28 nM T26623 C5IUX8 9814948 IC50 = 175 nM T26623 CL54TS 9814983 IC50 = 73 nM T26623 CIP84H 9819307 IC50 = 9 nM T26623 C5S8QT 9819308 IC50 = 1000 nM T26623 CS2VA9 9821758 IC50 = 99 nM T26623 C7Q2DN 9822496 IC50 = 100 nM T26623 CP37YD 9822749 IC50 = 3200 nM T26623 CP1M9D 9822861 IC50 = 8 nM T26623 CY84QK 9825086 IC50 = 25 nM T26623 C75IQH 9835612 IC50 = 280 nM T26623 CWZ13A 9836039 IC50 = 26 nM T26623 CRM4X5 9836072 IC50 = 360 nM T26623 CN8P1W 9836100 IC50 = 190 nM T26623 C5HD1Y 9836690 IC50 = 52 nM T26623 C5OCI3 9843574 IC50 = 11 nM T26623 C34ICB 9844233 IC50 = 5 nM T26623 C5E2RH 9844475 IC50 = 9 nM T26623 CUPN78 9846667 IC50 = 53 nM T26623 C5QJT6 9847444 IC50 = 30 nM T26623 CBLE73 9847475 IC50 = 52 nM T26623 CUS09M 9851899 IC50 = 4400 nM T26623 C0FGX3 9852086 IC50 > 200000 nM T26623 CN5IR4 9865185 IC50 = 163 nM T26623 CF2YU1 9866031 IC50 = 8 nM T26623 CGR1S9 9868478 IC50 = 100 nM T26623 CO3HT5 9874662 IC50 = 5700 nM T26623 CP74VE 9878604 IC50 = 870 nM T26623 CFK52A 9878605 IC50 = 390 nM T26623 CSZ34C 9879533 IC50 = 55 nM T26623 C36GDI 9879534 IC50 = 50 nM T26623 C0BG9I 9886690 IC50 = 17 nM T26623 C38TYU 9887806 IC50 = 10 nM T26623 CX86BD 9890496 IC50 = 8 nM T26623 CRH0P1 9901538 IC50 = 72 nM T26623 CJ7AS1 9902298 IC50 = 44 nM T26623 C30RBD 9902539 IC50 = 55 nM T26623 CV5T2F 9902829 IC50 = 667 nM T26623 CYMG76 9909523 IC50 = 11 nM T26623 C4OF7E 9913118 IC50 = 12 nM T26623 C5Y2ED 9922689 IC50 = 1100 nM T26623 CGM93U 9930308 IC50 = 8 nM T26623 C6X7OU 9930309 IC50 = 8 nM T26623 CZU5F4 9930310 IC50 = 6 nM T26623 C7DZ2I 9930503 IC50 = 7 nM T26623 C8TQ1M 9950615 IC50 = 660 nM T26623 CA7PN1 9952329 IC50 = 10 nM T26623 C4OTJ0 9955624 IC50 = 14 nM T26623 COMP92 9965222 IC50 = 422 nM T26623 C17KWZ 9966368 IC50 = 3 nM T26623 C94LYK 9966745 IC50 = 500 nM T26623 C72JBQ 9966787 IC50 = 35 nM T26623 CH51ND 9967430 IC50 = 140 nM T26623 C2RF7W 9970648 IC50 = 73.2 nM T26623 C3M0XB 9996408 IC50 = 52 nM T26623 CL8YG5 10018563 IC50 = 37 nM T26623 C3FKC4 10021783 IC50 = 1778 nM T26623 C2BF4G 10022229 IC50 = 115 nM T26623 C45TBJ 10023245 IC50 = 7943 nM T26623 C9VX0B 10042953 IC50 = 282 nM T26623 CAE21W 10043211 IC50 = 5623 nM T26623 CUW28C 10047003 IC50 = 1778 nM T26623 C1PU8F 10047735 IC50 = 190 nM T26623 CD58EL 10083644 IC50 = 2200 nM T26623 CQP3F8 10090285 IC50 = 1122 nM T26623 C15PXG 10095612 IC50 = 63 nM T26623 CTI26V 10098048 IC50 > 193500 nM T26623 CQR74M 10126802 IC50 > 100000 nM T26623 CS08XC 10133006 IC50 = 5 nM T26623 C28QWP 10150441 IC50 > 100000 nM T26623 CO23MY 10194147 IC50 > 100000 nM T26623 CS7A1W 10221192 IC50 = 49.3 nM T26623 CJ0EL5 10297924 IC50 = 13 nM T26623 CIFH75 10314257 IC50 = 46 nM T26623 CGXU05 10316809 IC50 = 4467 nM T26623 CBU2N9 10342270 IC50 = 226.6 nM T26623 CEA39F 10389369 IC50 = 12000 ug.mL-1 T26623 CD7Q2I 10402114 IC50 = 78.2 nM T26623 C9W0UP 10405318 IC50 = 1778 nM T26623 CSO29N 10407275 IC50 = 411 nM T26623 CEO91X 10409908 IC50 = 708 nM T26623 C2VR6L 10412732 IC50 = 144.1 nM T26623 CO9J2X 10424810 IC50 = 390 nM T26623 CF0VK2 10469744 IC50 = 30 nM T26623 CZ0I6Y 10473927 IC50 = 2239 nM T26623 CX3DY6 10788966 IC50 = 25 ug.mL-1 T26623 CU03EO 10968945 IC50 = 25 nM T26623 CFS2N7 11154496 IC50 = 1000 nM T26623 C0PZY4 11161499 IC50 = 73000 nM T26623 CZQU30 11184397 IC50 = 38600 nM T26623 CRLF61 11215672 IC50 = 3200 nM T26623 CJ4LH2 11235618 IC50 = 130 nM T26623 C4O6WF 11279241 IC50 = 34 nM T26623 CW0L9O 11290748 IC50 = 55 nM T26623 C4ZU8V 11291292 IC50 = 690 nM T26623 CI87WC 11292212 IC50 = 1600 nM T26623 C47HLT 11308405 IC50 = 8900 nM T26623 CRZT28 11343202 IC50 = 5500 nM T26623 C3DM1B 11349802 IC50 = 8 nM T26623 CKOV78 11405564 IC50 = 10.7 nM T26623 C58EJR 11507553 IC50 = 140 nM T26623 CP2F6R 11530302 IC50 = 87 nM T26623 C2HL5R 11536536 IC50 = 257 nM T26623 C7EG4P 11544083 IC50 = 645 nM T26623 C4I0HJ 11551271 IC50 = 230 nM T26623 CS91HB 11565723 IC50 = 13 nM T26623 CH0Y3G 11583024 IC50 = 3981 nM T26623 CQZ72F 11587295 IC50 = 118 nM T26623 CF6HD7 11587582 IC50 = 160 nM T26623 C1P0SQ 11588370 IC50 = 23 nM T26623 C1WQK8 11595367 IC50 = 200 nM T26623 C0B5DT 11595525 IC50 = 92 nM T26623 CF4L2K 11609768 IC50 = 6 nM T26623 CB1IC2 11652491 IC50 = 450 nM T26623 C2XV7T 11666475 IC50 = 1400 nM T26623 C2HBR8 11674139 IC50 = 3800 nM T26623 CS0UL4 11682497 IC50 = 34 nM T26623 CBJM05 11703420 IC50 = 49 nM T26623 C73ASH 11716421 IC50 = 54 nM T26623 C0NIV1 11716825 IC50 = 190 nM T26623 C9TR3K 11739835 IC50 = 560 nM T26623 CL5CO8 11743455 IC50 = 19.4 nM T26623 CX43MP 11833216 IC50 = 150 nM T26623 CZH0L3 12398821 IC50 = 1000 nM T26623 C5P7GO 12399888 IC50 > 100000 nM T26623 CSC28I 12512363 IC50 = 4500 nM T26623 CDU6E7 12536181 IC50 = 580 nM T26623 CP6AX4 12536182 IC50 = 270 nM T26623 C10TQF 12536184 IC50 = 360 nM T26623 CW20JC 12536185 IC50 = 510 nM T26623 CYC76W 12536190 IC50 = 10700 nM T26623 CUR9N3 12855920 IC50 > 200000 nM T26623 CAG9M1 13676777 IC50 = 770 nM T26623 C8YIZ5 13676778 IC50 = 5000 nM T26623 CWDN80 13676782 IC50 = 280000 nM T26623 CLS5G4 13676784 IC50 = 830 nM T26623 C72VBD 13676785 IC50 = 100000 nM T26623 CQP65A 13676786 IC50 = 160000 nM T26623 C79PXB 13676787 IC50 = 110000 nM T26623 CAU34B 13676788 IC50 = 210 nM T26623 C65LZV 13676789 IC50 = 760 nM T26623 CO6V9K 13676790 IC50 = 2700 nM T26623 C2MOL4 13850057 IC50 = 140 nM T26623 CN9UQ5 13850062 IC50 = 80 nM T26623 C5CH0S 13850064 IC50 = 820 nM T26623 CW8F2N 13850066 IC50 = 190 nM T26623 C4S1IV 13850068 IC50 = 200 nM T26623 CT15HV 13850074 IC50 = 29400 nM T26623 C2SI7K 13850075 IC50 = 910 nM T26623 CX38SO 13850077 IC50 = 3460 nM T26623 CQTF85 13850078 IC50 = 620 nM T26623 CNA35S 13850095 IC50 = 14800 nM T26623 CO0NY2 13850097 IC50 = 1670 nM T26623 C7VHK6 13850099 IC50 = 8220 nM T26623 C7RE1A 13850103 IC50 = 1000 nM T26623 CGI9P2 13850105 IC50 = 1180 nM T26623 C2BXK7 13850107 IC50 = 5160 nM T26623 CV4I6H 13850109 IC50 = 1630 nM T26623 C63WFH 13850113 IC50 = 240 nM T26623 CBPT07 13850115 IC50 = 110 nM T26623 C30IXB 13850117 IC50 = 90 nM T26623 CR21QZ 13850119 IC50 = 3320 nM T26623 C1E4BK 13850121 IC50 = 13100 nM T26623 C1PEW7 13850123 IC50 = 5700 nM T26623 C5Y3LQ 13850125 IC50 = 780 nM T26623 CBSQ65 13850127 IC50 = 70 nM T26623 C2D9CX 13850133 IC50 = 250 nM T26623 C7D2RM 13850135 IC50 = 130 nM T26623 CE36UR 13850137 IC50 = 50 nM T26623 C54JPQ 13850139 IC50 = 120 nM T26623 CNJ21B 13850141 IC50 = 4500 nM T26623 CX3QI8 13850143 IC50 = 100 nM T26623 CRGZ51 13850147 IC50 = 70 nM T26623 CMEF39 13850153 IC50 = 60 nM T26623 CRD91L 13850156 IC50 = 400 nM T26623 CZP71N 13953806 IC50 > 100000 nM T26623 C9WM0H 14109406 IC50 > 195300 nM T26623 CLB58T 14176152 IC50 = 112000 nM T26623 C2IA7B 14183548 IC50 = 1400 nM T26623 CHQ17F 14193987 IC50 = 119200 nM T26623 CZ7X4Q 14229968 IC50 = 56 nM T26623 CDV4H3 14229969 IC50 = 770 nM T26623 CKW6O0 14229970 IC50 = 100 nM T26623 C4SA3B 14229971 IC50 = 4500 nM T26623 CE2Q8H 14229972 IC50 = 64 nM T26623 CI8LN7 14229973 IC50 = 860 nM T26623 C4Q0RN 14229974 IC50 = 94 nM T26623 C62EAZ 14229975 IC50 = 4500 nM T26623 CKC49O 14229976 IC50 = 800 nM T26623 CM03PQ 14229977 IC50 = 1800 nM T26623 CAB7H2 14229978 IC50 = 360 nM T26623 C9Y4VF 14229979 IC50 = 220 nM T26623 CZU30F 14229980 IC50 = 400 nM T26623 CYC38H 14229981 IC50 = 59 nM T26623 C8V0SP 14229982 IC50 = 240 nM T26623 CBYA03 14229984 IC50 = 140 nM T26623 C5DOF4 14229985 IC50 = 42 nM T26623 C6EHA7 14229986 IC50 > 100000 nM T26623 C5BA6Y 14229987 IC50 > 100000 nM T26623 CQH05K 14229988 IC50 = 280 nM T26623 CT2VG9 14229989 IC50 = 310 nM T26623 CR18CH 14229990 IC50 = 3400 nM T26623 CZ13MC 14229994 IC50 = 72 nM T26623 C8CES3 14229997 IC50 = 74 nM T26623 CF5LM6 14230004 IC50 = 800 nM T26623 CVX28G 14230005 IC50 = 390 nM T26623 C1AZE8 14282455 IC50 = 560 nM T26623 COW37L 14371712 IC50 = 890 nM T26623 C7MLT9 14371713 IC50 = 7.5 nM T26623 CARK04 14371714 IC50 = 3090 nM T26623 C40VRP 14371716 IC50 = 950 nM T26623 CQDH02 14371717 IC50 = 7220 nM T26623 C31SHR 14389411 IC50 = 2200 nM T26623 CDTW54 14422820 Ki = 6800 nM T26623 CC1L9K 14422821 Ki = 5300 nM T26623 CML76V 14458620 IC50 = 680 nM T26623 CZYE18 14458621 IC50 = 58 nM T26623 C7CR0N 14458623 IC50 = 100 nM T26623 CQW25Y 14458649 IC50 = 6200 nM T26623 CYRL92 14458650 IC50 = 33 nM T26623 CI3T2S 14458654 IC50 = 30 nM T26623 CM9IY8 14458658 IC50 = 35 nM T26623 CEQM34 14458659 IC50 = 4.6 nM T26623 C31WBF 14458660 IC50 = 110 nM T26623 C43MPU 14458662 IC50 = 65 nM T26623 CZ79ME 14519545 IC50 = 6.3 nM T26623 CC34LV 14519546 IC50 = 460 nM T26623 C85DNA 14677893 IC50 = 17 nM T26623 CBE1H6 14773403 IC50 = 390 nM T26623 CB5XH3 14773437 IC50 = 970 nM T26623 C6VT9W 14773439 IC50 = 11300 nM T26623 CU0Y9B 14773441 IC50 = 400 nM T26623 C5E6JO 14773443 IC50 = 1860 nM T26623 C2VM6J 14773445 IC50 = 14800 nM T26623 CQ8E4C 14773447 IC50 = 5420 nM T26623 C4KP3C 14783857 IC50 = 1130 nM T26623 C1AZ7P 14792090 IC50 > 100000 nM T26623 C26QTM 14810637 IC50 = 3.1 nM T26623 CA0CU7 14810645 IC50 = 87 nM T26623 C57VTO 14810714 IC50 = 19 nM T26623 CZ3VQ2 14810715 IC50 = 2 nM T26623 C29SOV 14810716 IC50 = 3.5 nM T26623 CQPN60 14810717 IC50 = 25 nM T26623 CT2QL9 14810718 IC50 = 100 nM T26623 C4TA6H 14810719 IC50 = 100 nM T26623 CR2J9D 14810720 IC50 = 6.9 nM T26623 CLD26T 14810721 IC50 = 7.1 nM T26623 CX4YG2 14810722 IC50 = 26 nM T26623 C5Q6XW 14810723 IC50 = 41 nM T26623 C5DKA8 14810724 IC50 = 230 nM T26623 CLW0A8 14810725 IC50 = 60 nM T26623 CAPD90 14810726 IC50 = 4300 nM T26623 CD5V3M 14810727 IC50 = 1700 nM T26623 CNTS30 14810728 IC50 = 76 nM T26623 CS23AC 14810729 IC50 = 26 nM T26623 CKX3H5 14810730 IC50 = 3.1 nM T26623 CPJ4L9 14810733 IC50 = 320 nM T26623 C0L7PZ 14810734 IC50 = 1000 nM T26623 CUM4S0 14810735 IC50 = 4200 nM T26623 C9RFT4 14810736 IC50 = 3200 nM T26623 CUS3X8 14810737 IC50 = 1 nM T26623 C2WGS7 14810738 IC50 = 15 nM T26623 CKJ4Q9 14810739 IC50 = 10 nM T26623 C3VXR7 14810740 IC50 = 10 nM T26623 C9I0UH 14810741 IC50 = 100 nM T26623 COZ97G 14810742 IC50 = 510 nM T26623 CO2Y7U 14810743 IC50 = 68 nM T26623 C4Y2WS 14810744 IC50 = 110 nM T26623 C9J4OX 14810745 IC50 = 420 nM T26623 C75QGC 14810746 IC50 = 2300 nM T26623 C58PHC 14810747 IC50 = 120 nM T26623 C2Q6OF 14810748 IC50 = 4300 nM T26623 C2HT3U 14810749 IC50 = 320 nM T26623 CA7R9V 14810750 IC50 = 170 nM T26623 CL38IA 14810751 IC50 = 5 nM T26623 CF9GT0 14810752 IC50 = 20 nM T26623 C9IK3W 14810753 IC50 = 6.2 nM T26623 C40UQA 14810754 IC50 = 5 nM T26623 C2JYP4 14810755 IC50 = 100 nM T26623 CTF84S 14810756 IC50 = 620 nM T26623 C7RLO5 14810757 IC50 = 94 nM T26623 CLNX16 14810758 IC50 = 1400 nM T26623 CKF48Y 14810759 IC50 = 5.9 nM T26623 C6YRK1 14810760 IC50 = 660 nM T26623 CEF65Y 14810761 IC50 = 700 nM T26623 CRO34P 14810762 IC50 = 10 nM T26623 C9BK4I 14810763 IC50 = 4 nM T26623 CZ79WI 14810764 IC50 = 30 nM T26623 C1BD3A 14810765 IC50 = 15 nM T26623 CX2BL3 14810766 IC50 = 34 nM T26623 CX0MS1 14810767 IC50 = 690 nM T26623 C5B3FD 14810768 IC50 = 12 nM T26623 CLJW51 14810769 IC50 = 33 nM T26623 C5-OCT-02 14810770 IC50 = 46 nM T26623 C1O9JK 14810771 IC50 = 420 nM T26623 C0UB7Y 14810772 IC50 = 27 nM T26623 CO83HP 14810773 IC50 = 26 nM T26623 CRP18V 14810774 IC50 = 28 nM T26623 CCZ8E1 14810775 IC50 = 110 nM T26623 CR90YE 14810776 IC50 = 110 nM T26623 C9WA0B 14810777 IC50 = 12 nM T26623 CBM6U0 14810778 IC50 = 18 nM T26623 C68AUX 14810779 IC50 = 10 nM T26623 CAOC87 14810780 IC50 = 300 nM T26623 C3RP7X 14810781 IC50 = 42 nM T26623 CB24OI 14810782 IC50 = 1800 nM T26623 CJIR75 14810784 IC50 = 81 nM T26623 CJ56TX 14810785 IC50 = 43 nM T26623 C80FVP 14810788 IC50 = 5700 nM T26623 C4V9PC 14810789 IC50 > 100000 nM T26623 C45WGU 14810790 IC50 > 100000 nM T26623 CX6BI0 14820254 IC50 = 290 nM T26623 C5AL7X 14820306 IC50 = 760 nM T26623 CRY34Q 14852845 IC50 > 100000 nM T26623 C7LNY0 14852846 IC50 > 100000 nM T26623 CO3WN2 15035552 IC50 > 100000 nM T26623 CCE87Q 15074167 IC50 = 4000 nM T26623 C9P7VL 15074168 IC50 > 100000 nM T26623 CQM9B5 15074169 IC50 = 1000 nM T26623 C70SEK 15133803 IC50 = 2200 nM T26623 C8O1AE 15133804 IC50 = 1100 nM T26623 C0HL8A 15133805 IC50 = 3200 nM T26623 CIQB85 15133806 IC50 = 660 nM T26623 CX79PS 15133807 IC50 = 4500 nM T26623 CY4BL0 15133808 IC50 = 8200 nM T26623 CNBZ25 15133809 IC50 = 460 nM T26623 CG1MA8 15133810 IC50 = 34 nM T26623 CB2VH8 15133811 IC50 = 10000 nM T26623 C54VCR 15133812 IC50 = 670 nM T26623 C93SQV 15133813 IC50 = 37 nM T26623 CO4X2B 15133815 IC50 = 59000 nM T26623 CTPE31 15133816 IC50 = 160 nM T26623 C7CNF3 15133817 IC50 < 10 nM T26623 C4QB8K 15133818 IC50 = 23 nM T26623 C7UR8B 15133819 IC50 = 6.5 nM T26623 C1PCI3 15133820 IC50 = 6.4 nM T26623 C85HNK 15133821 IC50 = 220 nM T26623 CCGX79 15133822 IC50 = 470 nM T26623 CQE24V 15133823 IC50 = 4600 nM T26623 CK53UO 15133824 IC50 = 19 nM T26623 CV5I7U 15133825 IC50 = 630 nM T26623 C8LP3Q 15133826 IC50 = 240 nM T26623 CNX93T 15133827 IC50 = 156 nM T26623 C3JC0G 15133828 IC50 = 28 nM T26623 CK5T8X 15133829 IC50 = 470 nM T26623 CSJ07R 15133830 IC50 = 89 nM T26623 C4JDP7 15133831 IC50 = 78 nM T26623 CND8U9 15133832 IC50 = 27 nM T26623 CRNF81 15133833 IC50 = 31 nM T26623 CLD6Q2 15133834 IC50 = 540 nM T26623 C1O8LX 15133835 IC50 = 3.2 nM T26623 CJ3NB7 15133836 IC50 = 32 nM T26623 CU7I5S 15133837 IC50 = 6100 nM T26623 CT27IF 15133838 IC50 = 3000 nM T26623 CHU92E 15133839 IC50 = 120 nM T26623 CGK3E8 15133840 IC50 = 110 nM T26623 CN6JA7 15133841 IC50 = 150 nM T26623 CG8OB4 15133842 IC50 = 250 nM T26623 C1J0GL 15133843 IC50 = 1000 nM T26623 CR3K1A 15133844 IC50 = 2200 nM T26623 CT5D3U 15133845 IC50 = 420 nM T26623 C60IVD 15133846 IC50 = 150 nM T26623 CY7HU8 15133847 IC50 = 4200 nM T26623 C8ZR2L 15133848 IC50 = 870 nM T26623 C1D6LI 15133854 IC50 = 200 nM T26623 CN4G5E 15133855 IC50 = 170 nM T26623 COZ2H6 15133858 IC50 = 3100 nM T26623 CFUD60 15669766 IC50 < 10 nM T26623 CJ90TN 15669767 IC50 = 41 nM T26623 C8GK0B 15669768 IC50 = 26 nM T26623 CVUW18 15669769 IC50 = 2.1 nM T26623 C3SHA6 15669783 IC50 = 340 nM T26623 C8C2GI 15669784 IC50 < 10 nM T26623 CX75LE 15669785 IC50 = 18 nM T26623 CSX03W 15669786 IC50 <= 10 nM T26623 CXGE80 15669787 IC50 = 3.2 nM T26623 CV03OT 15669788 IC50 = 3.3 nM T26623 C3FHR1 15669789 IC50 = 32 nM T26623 CY2B8H 15669790 IC50 = 4 nM T26623 CZE1S6 15669791 IC50 = 420 nM T26623 CU34FZ 15669792 IC50 = 46 nM T26623 C18ADR 15708693 Ki = 4700 nM T26623 C6JP1K 15708694 Ki = 3100 nM T26623 C5ZAO3 15708695 Ki = 1300 nM T26623 C6Y1XR 15708696 Ki = 2500 nM T26623 CDC06Y 15708698 Ki = 310 nM T26623 C53TXR 15708699 Ki = 4300 nM T26623 CG5U9D 15708700 Ki = 2800 nM T26623 CU4OE1 15708701 Ki = 9700 nM T26623 C9UX7Q 15713958 IC50 = 2200 nM T26623 C2NS4A 15713959 IC50 = 19 nM T26623 C2E7JP 15713960 IC50 = 13 nM T26623 CV8U5K 15713961 IC50 = 440 nM T26623 CDM5S6 15713962 IC50 = 22 nM T26623 CJD3Q1 15713963 IC50 = 1100 nM T26623 CUO3X9 15713964 IC50 = 5900 nM T26623 CP3J4N 15713965 IC50 = 430 nM T26623 CIZ31F 15713966 IC50 = 2100 nM T26623 C3HE1P 15713967 IC50 = 4900 nM T26623 C5V2QW 15713969 IC50 = 200 nM T26623 C6GR7F 15713972 IC50 = 52 nM T26623 C8K7YC 15713973 IC50 = 50 nM T26623 CD3O2J 15727056 IC50 > 100000 nM T26623 CK4FB6 15733202 IC50 > 100000 nM T26623 CB6ZY1 15749969 IC50 = 281000 nM T26623 C71XUK 15749970 IC50 = 650 nM T26623 CIC5B6 15749971 IC50 = 95500 nM T26623 CG6C8O 15749972 IC50 = 43500 nM T26623 C6I4JZ 15749973 IC50 = 29400 nM T26623 CE39JD 15749974 IC50 = 600 nM T26623 CU34QM 15749976 IC50 = 11000 nM T26623 C3RS5K 15749977 IC50 = 11000 nM T26623 CHF1Q8 15749978 IC50 = 1140 nM T26623 C2BVM3 15750108 IC50 = 73 nM T26623 CNY0Q8 15750111 IC50 > 100000 nM T26623 CLI9B5 15750117 IC50 > 100000 nM T26623 CJ87YS 15750118 IC50 > 100000 nM T26623 CFU37X 15750119 IC50 = 2000 nM T26623 C5YD4V 15750120 IC50 = 6200 nM T26623 CPT16C 15750121 IC50 = 470 nM T26623 C71WTG 15750122 IC50 = 120 nM T26623 CF05BQ 15750123 IC50 = 260 nM T26623 CSM7O3 15750124 IC50 = 430 nM T26623 C9A6PG 15750125 IC50 = 130 nM T26623 CV70WT 15750127 IC50 = 480 nM T26623 CUC41L 16058629 IC50 = 30 nM T26623 CZ7P1I 16058630 IC50 = 6 nM T26623 C7UG2K 18468131 IC50 = 29 nM T26623 CS83QM 18468153 IC50 = 550 nM T26623 CQ71JG 18468166 IC50 = 7 nM T26623 C9B6GD 18468177 IC50 = 35 nM T26623 C1W0PV 19867112 IC50 = 37 nM T26623 CW27TQ 20055989 IC50 > 174700 nM T26623 C61MSD 20055991 IC50 > 194400 nM T26623 CZHU45 20055994 IC50 > 199200 nM T26623 C6HC5X 20291895 Ki = 400 nM T26623 CVH7N9 20308817 IC50 = 4000 nM T26623 CJKR07 21632954 IC50 > 189400 nM T26623 CK3U8M 21778114 IC50 = 0.11 ug.mL-1 T26623 C54IUM 21778115 IC50 = 0.4 ug.mL-1 T26623 CBJ3S1 21778116 IC50 = 0.25 ug.mL-1 T26623 C27BJH 21778117 IC50 = 0.4 ug.mL-1 T26623 C3H9CF 22093457 IC50 = 176 nM T26623 C8PU4J 24829377 IC50 = 741 nM T26623 CQ7DP2 24853736 IC50 = 1840 nM T26623 C01QNF 25014795 IC50 = 18200 nM T26623 C4QA6B 25761582 IC50 = 139 nM T26623 CVR78I 40466856 IC50 = 40000 nM T26623 C17PAG 42630080 IC50 = 1300 nM T26623 C7Q4XJ 42641743 IC50 = 31000 nM T26623 CAJ38Q 42641856 IC50 = 220 nM T26623 CY64IP 42641966 IC50 = 230 nM T26623 CX40IQ 42642081 IC50 = 200 nM T26623 C8DQ4J 43358934 IC50 = 42700 nM T26623 CF2G1L 44273340 IC50 = 140 nM T26623 CFA2J8 44273341 IC50 = 37 nM T26623 C6O7DU 44273392 IC50 = 26 nM T26623 CLN8O2 44298114 IC50 = 500 nM T26623 CZ84FG 44298252 IC50 = 6450 nM T26623 CSZF40 44305972 IC50 > 100000 nM T26623 CR40FP 44308834 IC50 = 570 nM T26623 C9K0DQ 44309003 IC50 = 1630 nM T26623 CZQ02C 44309018 IC50 = 2670 nM T26623 C85NIZ 44309019 IC50 = 360 nM T26623 CZ5K6L 44309072 IC50 = 1920 nM T26623 C34CPM 44309111 IC50 = 7650 nM T26623 CP62XH 44361448 IC50 = 720 nM T26623 CR9K1Y 44366031 IC50 = 25000 nM T26623 C9UTX4 44381246 IC50 = 3200 nM T26623 CP3JG2 44381460 IC50 = 7100 nM T26623 CRAB75 44381461 IC50 = 4300 nM T26623 CJ3S5V 44558965 IC50 = 25 ug.mL-1 T26623 CPV5W0 44558966 IC50 = 25 ug.mL-1 T26623 C6OBA9 44559090 IC50 = 25 ug.mL-1 T26623 C9XIW4 44590218 IC50 = 750 nM T26623 C34YPR 44724736 IC50 = 10.7 nM T26623 C90NLX 46853755 IC50 = 172 nM T26623 CR1JF6 46887680 IC50 > 200000 nM T26623 CU7ST1 51346826 IC50 > 50000 nM T26623 CMC96T 51370454 IC50 > 10000 nM T26623 C8B4DO 52918075 IC50 = 220 nM T26623 C1FCD5 52918076 IC50 = 400 nM T26623 CLT70X 52982948 IC50 = 0.66 nM T26623 CZ2UG1 53316850 IC50 = 169.82 nM T26623 C1OJ0M 53316888 IC50 > 50000 nM T26623 CG79XF 53316889 IC50 > 50000 nM T26623 CV90RX 53319308 IC50 = 900 nM T26623 CPD1Q7 53322999 IC50 = 1930 nM T26623 CZD9L1 53324788 IC50 = 60 nM T26623 C8LGY1 53325889 IC50 = 1620 nM T26623 CP2Q8Y 53373330 IC50 = 5900 nM T26623 CM7OL5 53373331 IC50 = 4200 nM T26623 CZ31JH 53373332 IC50 = 10000 nM T26623 CE5A8I 54580480 IC50 > 200000 nM T26623 CAS91K 54682930 IC50 > 400000 nM T26623 CS8R0Z 54716566 IC50 = 5500 nM T26623 C94NVX 56591766 IC50 = 170 nM T26623 C91TGZ 56591768 IC50 = 4900 nM T26623 CB5V7P 56838291 IC50 = 150 nM T26623 CLO87D 56964583 IC50 = 27700 nM T26623 C34IBM 57328732 IC50 = 41000 nM T26623 C1P8SB 57328733 IC50 = 1100 nM T26623 C94NWO 57328735 IC50 = 7200 nM T26623 C86OHG 57328736 IC50 = 9500 nM T26623 C6QCJ0 57328737 IC50 = 7300 nM T26623 CVF3D1 57328738 IC50 = 3200 nM T26623 CEU25K 57328803 IC50 = 11000 nM T26623 CWK8Q7 57328804 IC50 = 6900 nM T26623 CT5F4I 57328805 IC50 = 11000 nM T26623 CO4N2H 57391537 IC50 > 189400 nM T26623 C3CO5H 57391659 IC50 = 190 nM T26623 CO6C3W 57391660 IC50 = 200 nM T26623 C3Q6RC 57393486 IC50 = 320 nM T26623 CK1ET9 57393918 IC50 = 2239 nM T26623 C1M0LS 57394809 IC50 = 6100 nM T26623 CS4RY2 57395022 IC50 > 183900 nM T26623 CK3ZF7 57395128 IC50 = 350 nM T26623 C63FCJ 57395129 IC50 = 190 nM T26623 CSIK32 57395208 IC50 = 1700 nM T26623 C8BOQ9 57396771 IC50 = 43800 nM T26623 CIX6H9 57396988 IC50 = 48600 nM T26623 C3WET7 57398539 IC50 > 183900 nM T26623 CS10LY 57398744 IC50 = 14000 nM T26623 C0QFN8 57400324 IC50 = 1800 nM T26623 CI05FH 57400872 IC50 = 3160 nM T26623 CCE5O6 57402147 IC50 = 22800 nM T26623 CY38WL 57402652 IC50 = 3162 nM T26623 CC26MG 57403756 IC50 > 174200 nM T26623 CKE78V 57403960 IC50 = 240 nM T26623 CO75NL 68011817 IC50 = 150 nM T26623 C4ZC7T 70695255 IC50 = 350 nM T26623 C9O2BS 71716678 IC50 = 100000 nM T26623 CGJM90 71718524 IC50 > 100000 nM T26623 C7Z5IO 72205881 IC50 > 10000 nM T26623 CKP3V9 72205882 IC50 > 10000 nM T26623 CTBL48 73055653 IC50 = 9000 nM T26623 CD96TP 76308360 IC50 = 6.18 nM T26623 CIF41J 76315831 IC50 = 13.4 nM T26623 CRW7B4 76319237 IC50 = 4.17 nM T26623 C5M4RN 76322885 IC50 = 39.1 nM T26623 CC0IM2 76326455 IC50 = 6.14 nM T26623 CD5A8T 76330077 IC50 = 1.32 nM T26623 CVB5I0 76333726 IC50 = 1.19 nM T26623 CECP92 90643583 IC50 = 228 nM T26623 CZ39XP 90643584 IC50 = 64 nM T26623 C2EXC3 97686398 IC50 = 104 nM T26623 C9A0GL 101937482 IC50 = 23000 nM T26623 CH8K9G 102258078 IC50 = 650 nM T26623 CX7TF9 102258079 IC50 = 240 nM T26623 CTY9D5 102258080 IC50 = 3200 nM T26623 C9V5IP 102258081 IC50 = 130 nM T26623 C4UZ1A 110667198 IC50 > 10000 nM T26623 CO73US 117058579 Ki = 66.1 nM T26623 C6I8AH 118708725 IC50 = 98 nM T26623 CR61CY 118711690 IC50 > 200000 nM T26623 CAT4K8 118720624 IC50 > 200000 nM T26623 CH0W4M 122174240 IC50 = 21700 nM T26623 CDBY61 124922745 IC50 = 364 nM T26623 CZ8IP9 132520924 IC50 = 100 nM T26623 CN3ZA9 132917086 IC50 > 100000 nM T26623 C3F6WD 134133107 IC50 = 109000 nM T26623 C3QHI5 134142061 IC50 = 540 nM T26623 C5B1WP 134152926 IC50 = 310 nM T26623 C92VFA 135450383 IC50 = 34 nM T26623 CUZ13N 135483714 Ki = 7800 nM T26623 CW09LA 135487739 Ki = 9300 nM T26623 CH1JX2 135512117 IC50 = 11 nM T26623 CY9O5S 135512118 IC50 = 21 nM T26623 CW2Q3O 135512119 IC50 = 36 nM T26623 CP9U1V 135535745 Ki = 150 nM T26623 C0PEH4 135631466 IC50 = 34 nM T26623 CO9WT8 135631469 IC50 = 26 nM T26623 C26CWR 136219384 IC50 = 28 nM T26623 CI2K1G 136219385 IC50 = 24 nM T26623 CPM7Y9 136219386 IC50 = 25 nM T26623 C4K1AD 136229863 IC50 = 24 nM T26623 C6TI1F 136229864 IC50 = 19 nM T26623 C45AXN 136229867 IC50 = 12 nM T26623 C7RWY1 136229868 IC50 = 20 nM T26623 C6S1BG 136229869 IC50 = 6.7 nM T26623 C1R2YW 136229870 IC50 = 28 nM T26623 C2O0QF 136229872 IC50 = 27 nM T26623 CRB32G 136229881 IC50 = 20 nM T26623 CLQD65 136229882 IC50 = 29 nM T26623 CDZ47E 136229883 IC50 > 10000 nM T26623 CVBI32 137633456 IC50 = 320 nM T26623 CQI6H0 137636103 IC50 = 340 nM T26623 CJ9AP8 137636440 IC50 = 200 nM T26623 C08OEH 137639882 IC50 = 314 nM T26623 CQ4V6K 137639883 IC50 = 180 nM T26623 CHBZ93 137642578 IC50 = 15 nM T26623 C4UE9D 137642579 IC50 = 277 nM T26623 C2U3LN 137646926 IC50 = 9500 nM T26623 CR10SV 137646927 IC50 = 204 nM T26623 C61YPT 137647031 IC50 = 390 nM T26623 CJWD24 137660885 IC50 = 220 nM T26623 C6I0ZF 154732246 IC50 = 66 nM T26623 CRA6K8 155512220 IC50 = 20 nM T26623 C5LN0V 155518931 IC50 = 22200 nM T26623 CVI14S 155519450 Ki = 16 nM T26623 C2J7TE 155521721 IC50 = 560 nM T26623 CY9GB3 155522284 IC50 = 5840 nM T26623 C1XAK0 155523413 IC50 = 37720 nM T26623 CDY1Q8 155523913 IC50 = 40150 nM T26623 CF3W1J 155525280 IC50 = 323 nM T26623 CAL2P9 155525427 IC50 = 46 nM T26623 C4BVF8 155526535 Ki = 6.2 nM T26623 CSD79K 155526576 IC50 = 370 nM T26623 C2LGP9 155526813 IC50 = 6210 nM T26623 CCKW61 155529053 IC50 = 6150 nM T26623 C8IY4M 155536411 IC50 = 5660 nM T26623 CC1MA3 155537004 IC50 = 5020 nM T26623 CV1J9E 155539348 IC50 = 8020 nM T26623 C6C7ZQ 155540504 IC50 = 1410 nM T26623 C46QNR 155542010 IC50 = 24250 nM T26623 C2SXD8 155542498 IC50 = 34500 nM T26623 C31GUV 155547724 IC50 = 1800 nM T26623 CCA31E 155550245 IC50 = 640 nM T26623 C0Z4CP 155556329 IC50 = 930 nM T26623 CP89ZC 155558498 IC50 = 11660 nM T26623 C02ZPG 155564598 IC50 = 10840 nM T26623 CM8RN1 155564684 IC50 = 5720 nM T26623 D00EPD 9921581 IC50 = 170 nM T26623 D00KCB 449157 IC50 = 11000 nM T26623 D00RIX 5280443 IC50 = 11900 nM T26623 D00VHG 1944 IC50 = 108 nM T26623 D01BKS 9918693 IC50 > 200000 nM T26623 D01BZE 73659 IC50 = 72000 nM T26623 D01KKU 5281894 IC50 = 12300 nM T26623 D01UYI 5281607 IC50 = 7780 nM T26623 D02AAH 9878572 IC50 = 380 nM T26623 D02HCQ 1794427 IC50 = 300 nM T26623 D02JEZ 5281426 IC50 = 22900 nM T26623 D02WZA 10902449 IC50 = 450 nM T26623 D03LRQ 10398922 IC50 = 2400 nM T26623 D03NPA 471002 IC50 > 193500 nM T26623 D03YBR 23647383 IC50 = 600 nM T26623 D03ZMQ 323 IC50 > 500000 nM T26623 D05PTT 5281792 IC50 = 3910 nM T26623 D05QOR 5280460 IC50 = 74400 nM T26623 D06YGF 5281787 IC50 = 570 nM T26623 D06YQS 9943009 IC50 = 540 nM T26623 D07DJS 5280459 IC50 = 150 nM T26623 D07JEY 448658 IC50 = 11 nM T26623 D07LUJ 64945 IC50 = 41000 nM T26623 D07XXK 10267673 IC50 = 2200 nM T26623 D08BFU 5282102 IC50 = 60500 nM T26623 D08JEI 11673647 IC50 = 360 nM T26623 D09OWC 5373936 IC50 = 40830 nM T26623 D09PNQ 751 IC50 = 10 nM T26623 D0A1CM 5281855 IC50 = 200 nM T26623 D0A2FM 9856809 IC50 = 5000 nM T26623 D0AU0M 637542 IC50 = 140 nM T26623 D0E0RW 69894 IC50 = 56200 nM T26623 D0FJ7G 4369325 IC50 = 30 nM T26623 D0G3TK 5280863 IC50 = 10000 nM T26623 D0IB8C 22424988 IC50 = 1900 nM T26623 D0LC7K 119034 IC50 = 34000 nM T26623 D0O9KV 9901432 IC50 = 210 nM T26623 D0OC4B 5357479 IC50 = 2400 nM T26623 D0OZ4C 11701437 IC50 = 600 nM T26623 D0P1ZM 9943757 IC50 = 150 nM T26623 D0P3AU 9921499 IC50 = 2000 nM T26623 D0Q7DJ 10742 IC50 = 172.1 ug.mL-1 T26623 D0R3MB 11807954 IC50 = 25 nM T26623 D0R7IJ 9943365 IC50 = 240 nM T26623 D0S9YX 5280373 IC50 = 127000 nM T26623 D0SJ2Q 10494 IC50 = 124000 nM T26623 D0SY2M 5281708 IC50 = 161800 nM T26623 D0T2QL 444539 IC50 = 68.1 ug.mL-1 T26623 D0T3PW 5281672 IC50 = 29000 nM T26623 D0U4BB 10748 IC50 = 67500 nM T26623 D0U4VL 5472440 IC50 = 23000 nM T26623 D0U8IF 10114 IC50 = 280000 nM T26623 D0V9EN 689043 IC50 = 32000 nM T26623 D0XD1Q 9856396 IC50 = 474 nM T26623 D0Y3TZ 370 IC50 = 97.3 ug.mL-1 T26623 D0Y7PW 11674065 IC50 = 350 nM T26623 D0YZ5G 5281416 IC50 = 67200 nM T77181 D03GET 4055 IC50 = 71000 nM T77181 CS9RO8 2729042 IC50 = 600 nM T77181 CM31XR 2891549 IC50 = 154000 nM T77181 CQA1Y4 2913480 IC50 = 123000 nM T77181 C0JS2N 2941245 IC50 = 103000 nM T77181 C3Z5CV 46830074 IC50 > 200000 nM T77181 C3P8EW 52940990 IC50 = 23000 nM T77181 CEW74T 52942184 IC50 = 47000 nM T77181 CU0H7T 52943029 IC50 = 17000 nM T77181 CA6BT2 52944213 IC50 = 25000 nM T77181 D0N6BC 950368 Ki = 100000 nM T39977 D0B8MZ 124246 IC50 = 6810 nM T39977 D0BQ8Y 5971 IC50 = 250 nM T39977 D0ZX2G 3598 Ki = 5550 nM T39977 D04KKT 4633677 IC50 = 7000 nM T39977 D07AOL 16741 IC50 = 16000 nM T39977 D0B1FE 3194 Ki = 570 nM T39977 CNI9Q6 853 IC50 = 15800 nM T39977 CT3IS2 2346 IC50 = 540 nM T39977 C30CLK 7673 IC50 = 11000 nM T39977 CAE87W 8106 IC50 = 17400000 nM T39977 CFG3Y9 17460 IC50 = 810 nM T39977 CL61DI 18170 IC50 > 100000 nM T39977 CCL54V 20559 IC50 = 1000 nM T39977 CIM58P 75815 IC50 = 1400 nM T39977 CT4WH9 75963 IC50 = 540 nM T39977 CG8V3C 114757 IC50 = 4200 nM T39977 CP46UJ 123197 IC50 = 700 nM T39977 CW5FK0 124881 IC50 = 1900 nM T39977 CPK92S 140257 IC50 = 1100 nM T39977 CLA4Y2 160602 IC50 > 100000 nM T39977 CQA6U5 520742 IC50 > 100000 nM T39977 CIC1N8 720432 IC50 = 21000 nM T39977 CJ0X7D 746669 Ki = 1600 nM T39977 CPA78N 755496 IC50 = 980000 nM T39977 CPFB08 763707 Ki = 6200 nM T39977 CL0U2D 764266 Ki = 26600 nM T39977 CE9PK0 794467 IC50 = 62100 nM T39977 C4S1KU 807516 IC50 = 85560 nM T39977 CIH1U5 833376 IC50 = 370 nM T39977 C3BF9K 866325 IC50 = 102120 nM T39977 CF3G8N 898930 IC50 = 6900 nM T39977 CNHO92 1105140 IC50 = 74490 nM T39977 C48MKW 1265466 IC50 = 45540 nM T39977 CN4A7B 1292657 IC50 = 22570 nM T39977 CA34NW 1327076 Ki = 348 nM T39977 CZ3GW0 1328188 Ki = 5141 nM T39977 C48YHR 1473456 IC50 = 300000 nM T39977 CK8PO4 1510388 IC50 = 4200 nM T39977 CE2R7Q 1519965 IC50 = 6200 nM T39977 CB9S5I 1752837 IC50 = 23060 nM T39977 C1WXK5 2202512 Ki = 4521 nM T39977 CA4BL3 2277207 IC50 = 9500 nM T39977 CI37FJ 2725942 Ki = 52 nM T39977 CE4X2Z 2727457 IC50 = 430000 nM T39977 CD8AY0 2737275 IC50 = 1500 nM T39977 CZGM75 2795371 IC50 = 2900 nM T39977 C5OM8W 2821653 IC50 = 60400 nM T39977 C3DX7F 3136927 IC50 = 3400 nM T39977 CCB05J 3748059 IC50 = 120800 nM T39977 C58FZC 5012755 IC50 = 530000 nM T39977 CU72RN 5288525 IC50 = 7000 nM T39977 CH85QC 5393173 Ki = 2900 nM T39977 C53DXS 5408870 Ki = 2100 nM T39977 CE4UF5 5413038 IC50 = 64200 nM T39977 CQ4IW2 5666318 Ki = 5800 nM T39977 CU06SR 6468009 IC50 = 18600 nM T39977 C4BKE8 6494116 IC50 = 730000 nM T39977 CZ9GO4 7015180 IC50 = 1100 nM T39977 CUB2M3 7174253 Ki = 113000 nM T39977 CE76SB 7221250 IC50 = 25770 nM T39977 CY8H9I 10442282 IC50 = 1200 nM T39977 CV7U8B 10538568 IC50 = 19700 nM T39977 CTO0U8 10847334 IC50 = 16700 nM T39977 CLHX93 11019761 IC50 = 29000 nM T39977 CZY5H7 12125208 IC50 = 750 nM T39977 C2RD1A 12622909 IC50 = 21000 nM T39977 CVT54A 13975638 IC50 = 5900 nM T39977 C2GD1A 14680579 IC50 = 38 nM T39977 C3SIU1 16007100 IC50 > 100000 nM T39977 CBOW60 17605128 IC50 = 1800 nM T39977 CVDQ34 18386401 Ki = 2600 nM T39977 CQ9H5O 20673360 Ki = 30900 nM T39977 CV4AP2 25181243 IC50 = 6500 nM T39977 CT3NB9 25241618 IC50 = 5600 nM T39977 CHA6W3 44182102 IC50 = 2800 nM T39977 CHO09B 44406772 IC50 = 8000 nM T39977 C4N5YX 44406779 IC50 = 30000 nM T39977 CTJ1D7 44580830 Ki = 1600 nM T39977 C94JYR 44613703 IC50 = 5100 nM T39977 C1MQ4S 44631884 IC50 = 10 nM T39977 C0B6KA 45268606 IC50 = 55000 nM T39977 CZ7P4U 45268613 IC50 = 12000 nM T39977 C1DHV8 45270292 IC50 > 100000 nM T39977 CLUK50 45270304 IC50 > 100000 nM T39977 CZ2VG7 45272022 IC50 = 32000 nM T39977 CM7QO9 45273787 IC50 = 100000 nM T39977 CIL02T 45273788 IC50 = 30000 nM T39977 CA4F1I 49847519 IC50 = 4800 nM T39977 CLR9D2 49863985 IC50 = 6000 nM T39977 CGLT17 50908752 IC50 = 750 nM T39977 CYBO20 50908753 IC50 = 2500 nM T39977 C12QAM 50908754 Ki = 37000 nM T39977 CI59ZN 52941336 IC50 = 970000 nM T39977 C8AP5V 52941421 IC50 = 2100 nM T39977 C7A8HQ 52942228 IC50 = 475000 nM T39977 CTGE28 52942373 IC50 = 70000 nM T39977 COGC30 52942624 IC50 = 1000000 nM T39977 C8PHT4 52942633 IC50 = 2900 nM T39977 CY1D2Z 52943617 IC50 = 32000 nM T39977 CHG60R 52943807 IC50 = 690000 nM T39977 CY0FL8 52945122 IC50 = 2500 nM T39977 CCM76J 52945126 IC50 = 26000 nM T39977 CYWH78 52946480 IC50 = 530000 nM T39977 CJH9B7 52947759 IC50 = 7.5 nM T39977 CDIC25 52948461 IC50 = 65000 nM T39977 CNR5X6 52949985 IC50 = 30000 nM T39977 C8V1MD 53363919 IC50 = 1000 nM T39977 CHV45O 53363920 IC50 = 6400 nM T39977 C6A7GJ 54122801 IC50 = 25200 nM T39977 CCU84Q 54588465 IC50 = 2800 nM T39977 CN9M4L 54588466 IC50 = 3100 nM T39977 C1DS6B 56659768 IC50 = 19000 nM T39977 CUWS73 56663237 IC50 = 8000 nM T39977 CGF6L9 56663240 IC50 = 5600 nM T39977 C9HNQ2 56663241 IC50 = 11000 nM T39977 C8FZS3 56663242 IC50 = 4800 nM T39977 CZRH46 56666676 IC50 = 5900 nM T39977 CH9OK1 56670099 IC50 = 4900 nM T39977 CS7Y6A 56673606 IC50 = 2400 nM T39977 CT59NF 56673607 IC50 = 1900 nM T39977 CUV59I 56673608 IC50 = 25000 nM T39977 C0LM9F 56676932 IC50 = 7900 nM T39977 C52JSO 56680240 IC50 = 5000 nM T39977 C3E2ND 56680246 IC50 = 8500 nM T39977 CK0T7S 56683572 IC50 = 2300 nM T39977 CQ80PH 56683580 IC50 = 6600 nM T39977 C4EN7R 56683581 IC50 = 6200 nM T39977 CD14PR 57392315 IC50 = 55300 nM T39977 C7EDZ2 57397608 IC50 = 11200 nM T39977 C2X0JR 57399362 IC50 = 37200 nM T39977 CN51OD 57402809 IC50 = 35400 nM T39977 CLN56X 71299360 IC50 = 6200 nM T39977 C15NYT 71299377 IC50 = 13500 nM T39977 C8ANC9 71460891 Ki = 270000 nM T39977 CP4L2I 71462587 Ki = 101000 nM T39977 CQZ6R0 84105919 IC50 = 7100 nM T39977 C58KCU 84105925 IC50 = 62000 nM T39977 CIP09N 90684376 Ki = 230 nM T39977 C63CXP 90684377 Ki = 200 nM T39977 CPIG49 91667574 Ki = 24 nM T39977 CTY98A 91667576 Ki = 14 nM T39977 C6XOI1 91971983 Ki = 300 nM T39977 CNM81O 118430419 Ki = 100 nM T39977 CR1ZL2 118430620 Ki = 1000 nM T39977 CPY3J6 118437635 Ki = 2000 nM T39977 C3LMU5 118731499 IC50 = 10400 nM T39977 CN17VP 118731500 IC50 > 100000 nM T39977 CAPY74 118731588 IC50 = 1200 nM T39977 CF28GK 122219230 Ki = 160 nM T39977 CDYM49 122219231 Ki = 74 nM T39977 CBM5V7 122457239 Ki = 48 nM T39977 CA5OB4 122457241 Ki = 363 nM T39977 C6FIZ7 122457316 Ki = 39 nM T39977 CTA8S1 122457321 Ki = 37 nM T39977 C0TA4U 122495069 Ki = 200 nM T39977 CP2EJ9 127046251 IC50 = 110 nM T39977 C3C8JK 131953495 Ki = 75 nM T39977 CYSF54 132473015 Ki = 510 nM T39977 C7LAM5 134133406 Ki = 260 nM T39977 CB6J8F 134135175 Ki = 147 nM T39977 C9NDR6 134140799 Ki = 530 nM T39977 C0OZ9Y 134142774 Ki = 360 nM T39977 CYC38Q 134145866 Ki = 1370 nM T39977 CNB4E8 134146410 Ki = 270 nM T39977 C72EZY 134155978 Ki = 144 nM T39977 CE2Y9H 135409923 IC50 = 15200 nM T39977 CC1N2R 135442230 IC50 = 70000 nM T39977 CBP7C0 135452431 IC50 = 43000 nM T39977 CSMX86 135480563 IC50 = 5500 nM T39977 CIGX15 135483672 Ki = 1500 nM T39977 CVI9T0 135484536 IC50 = 1650 nM T39977 CO56BU 135496292 IC50 = 10000 nM T39977 CX0Y2H 135501601 IC50 > 100000 nM T39977 C4B3VI 135502886 Ki = 550 nM T39977 CH4UE3 135510345 IC50 = 300000 nM T39977 C3F7DH 135510348 IC50 = 8000 nM T39977 C0K6FR 135510427 Ki = 280 nM T39977 C9H0NX 135512729 IC50 > 100000 nM T39977 CLO29N 135540733 Ki = 3100 nM T39977 CUMQ05 135542501 IC50 = 100000 nM T39977 CC6BD4 135544543 IC50 = 100000 nM T39977 CQ7O8V 135564896 IC50 = 13000 nM T39977 CISE20 135572086 IC50 = 7000 nM T39977 C3Y2OR 135581769 IC50 = 55000 nM T39977 C7KWB2 135616912 IC50 = 11000 nM T39977 CO8I1F 135616913 IC50 = 4000 nM T39977 C65SAZ 135616914 IC50 = 1300 nM T39977 CGBL45 135845046 IC50 = 1500 nM T39977 CV2DC3 135845047 IC50 = 750 nM T39977 CY5AC8 135857233 IC50 = 500 nM T39977 CPCT53 135908260 IC50 = 7000 nM T39977 CY8SH5 135965910 IC50 = 60000 nM T39977 CRUQ95 135965912 IC50 = 29000 nM T39977 C1S4XH 135965913 IC50 = 15000 nM T39977 CUF50Q 135965914 IC50 > 100000 nM T39977 C9YNZ8 135965940 IC50 = 48000 nM T39977 C7JNG5 135965945 IC50 > 100000 nM T39977 C4WLI1 135966018 IC50 = 60000 nM T39977 CZC40T 135966020 IC50 = 15000 nM T39977 CH65AJ 135966062 IC50 = 28000 nM T39977 CG4MX7 135966063 IC50 = 15000 nM T39977 C8GBY4 135966064 IC50 = 2000 nM T39977 CK12ZU 135973099 IC50 = 5000 nM T39977 C7CZ3A 135973104 IC50 = 24000 nM T39977 C17YVP 135973115 IC50 = 2500 nM T39977 C5S0GF 135993340 IC50 = 7000 nM T39977 C7HO1Z 135995954 Ki = 500 nM T39977 CT5ZC0 136036578 IC50 = 3000 nM T39977 C7ZGV8 136036584 IC50 = 3400 nM T39977 CN38YC 136036585 IC50 = 14500 nM T39977 CAJ8I6 136036586 IC50 = 7000 nM T39977 C6OBX4 136036592 IC50 = 113000 nM T39977 C53XCT 136036593 IC50 = 147000 nM T39977 CH4FT2 136036594 IC50 = 25000 nM T39977 CCV6R5 136042214 IC50 = 7300 nM T39977 C1L5NI 136042215 IC50 = 10200 nM T39977 CR8UH0 136043744 IC50 = 26000 nM T39977 CU6LW4 136043745 IC50 = 8500 nM T39977 CFC0P4 136043746 IC50 = 20000 nM T39977 CPT04L 136043748 IC50 > 100000 nM T39977 C97QYS 136043749 IC50 = 12000 nM T39977 CL6CO3 136043750 IC50 = 4000 nM T39977 CZSV23 136043751 IC50 = 6000 nM T39977 C8XB1J 136043753 IC50 = 10000 nM T39977 C8BNY1 136043754 IC50 = 8500 nM T39977 CRV2X8 136043755 IC50 = 10000 nM T39977 CIV5M0 136043766 IC50 = 550 nM T39977 C7HS3G 136043769 IC50 = 1100 nM T39977 CQH87O 136043770 IC50 = 6500 nM T39977 CQC1V5 136043773 IC50 = 3000 nM T39977 C81JEP 136102116 IC50 = 550 nM T39977 C9HD6M 136110958 IC50 = 50000 nM T39977 C9EU1T 136110959 IC50 > 50000 nM T39977 CWD9J6 136110960 IC50 = 10000 nM T39977 CNU3V4 136123459 IC50 = 25000 nM T39977 CROP52 136123460 IC50 = 50000 nM T39977 CR1F0E 136123461 IC50 = 20000 nM T39977 CB0WK5 136123462 IC50 > 100000 nM T39977 CS4N8U 136123500 IC50 = 19000 nM T39977 C7NK4G 136494499 IC50 = 1500 nM T39977 C40FJB 136961583 IC50 = 7000 nM T39977 CRF4P2 137224952 IC50 = 410 nM T39977 CH1XP7 137241594 Ki = 24000 nM T39977 C2HUI4 137349074 Ki = 90 nM T39977 CQ41XU 137640655 Ki = 1000 nM T39977 C9A3RE 139491193 Ki = 67 nM T39977 C6U9JM 145965166 Ki = 56 nM T39977 CQU4T5 145965652 IC50 = 7100 nM T39977 CCKD03 145967417 IC50 = 13000 nM T39977 CEM6F7 145967419 Ki = 2470 nM T39977 CN5PE8 145974041 IC50 = 8000 nM T39977 C3AMD8 145974507 IC50 = 21000 nM T39977 D01HJN 5289613 Ki = 7400 nM T39977 D03IWC 52950186 IC50 = 3400 nM T39977 D03QNS 5393176 Ki = 470 nM T39977 D04MZK 6403448 IC50 = 50 nM T39977 D05RSQ 52942744 IC50 = 1000 nM T39977 D07OLL 44406762 IC50 = 400 nM T39977 D08IXW 97536 IC50 = 3300000 nM T39977 D09BVA 5392139 Ki = 4300 nM T39977 D0A1CM 5281855 Ki = 1950 nM T39977 D0A5XY 1348789 IC50 = 2800 nM T39977 D0E1HP 75107 IC50 = 8100 nM T39977 D0J5DN 5284648 Ki = 38 nM T39977 D0O4BU 2202888 IC50 = 80 nM T39977 D0S0YQ 972361 IC50 = 1010 nM T39977 D0V4SG 1087842 IC50 = 500 nM T39977 D0W1JY 39763 IC50 = 40000 nM T39977 D0W1WF 817368 IC50 = 4500 nM T39977 D0X4IO 5350 IC50 = 2200 nM T39977 D0Y2OB 780029 IC50 = 3000 nM T39977 D0YY2W 870537 IC50 = 300 nM T18876 D06FEA 5280360 EC50 = 0.02 nM T18876 D0WL5V 9867642 Ki > 15200 nM T18876 D00HTY 5280363 IC50 = 4200 nM T18876 D00IQH 11677589 IC50 = 11.7 nM T18876 D00MZK 9911469 Ki > 10000 nM T18876 D00SOZ 44230999 IC50 > 10000 nM T18876 D01SHJ 56944705 IC50 = 7.5 nM T18876 D03YAS 9824353 EC50 = 0.01 nM T18876 D0G6EI 9890801 Ki > 3200 nM T18876 D0HJ5H 25209437 Ki = 3 nM T18876 D0K1EG 11508736 IC50 > 10000 nM T18876 D0M4TJ 44219292 Ki = 678 nM T18876 D0SP5V 49843471 IC50 > 10000 nM T18876 D0Y3LL 18376177 Ki > 3200 nM T18876 D0W2OT 5311035 Ki > 10000 nM T18876 D02RUO 9807448 Ki > 10000 nM T18876 D08QHS 11296282 IC50 = 8039 nM T18876 CZO8Y9 775693 IC50 = 2600 nM T18876 CNSZ97 786859 Ki = 420 nM T18876 COE84W 1144137 IC50 = 1000 nM T18876 CMNJ82 1351369 IC50 = 128 nM T18876 CANV86 1498200 Ki > 2700 nM T18876 C3LM8E 1498314 Ki > 2700 nM T18876 CLM8P6 2114670 Ki > 25000 nM T18876 C5IJ2D 2883793 IC50 = 4600 nM T18876 CIE7W0 3756926 IC50 = 460 nM T18876 C2XLU7 5311228 Ki = 2300 nM T18876 CO7N1Z 5311239 IC50 > 10000 nM T18876 C65ONU 6453527 EC50 = 200000 nM T18876 CZA41R 9808508 Ki > 100000 nM T18876 C6TA3N 9809136 Ki = 5000 nM T18876 CV24TI 9817292 Ki > 50000 nM T18876 C5WL7C 9821171 EC50 = 0.03 nM T18876 C5J8WP 9830442 Ki > 100000 nM T18876 CG3IS9 9830839 Ki = 46 nM T18876 COU85R 9863804 EC50 = 5 nM T18876 C97MIQ 9865111 Ki = 440 nM T18876 C6V1BA 9872741 Ki > 100000 nM T18876 CA2I4Z 9873528 Ki = 6000 nM T18876 CKMW12 9874010 Ki = 1100 nM T18876 C38DYF 9885106 Ki = 3.8 nM T18876 CF0HC5 9888589 IC50 > 10000 nM T18876 CFC8G4 9894720 Ki = 0.3 nM T18876 CA5N0K 9895436 Ki = 2400 nM T18876 CPCJ19 9907375 EC50 = 190 nM T18876 C7MA6V 9916766 Ki > 100000 nM T18876 CI8PZ7 9931112 EC50 = 19.95 nM T18876 CN2UX4 9938625 Ki = 13000 nM T18876 CICE70 9938626 Ki = 20000 nM T18876 C1KAC5 9938669 Ki = 7000 nM T18876 C6DQ3W 9938995 Ki > 100000 nM T18876 CWDT69 9939791 Ki = 4000 nM T18876 CWS81C 9944231 Ki = 6000 nM T18876 C4Q7RI 9953337 Ki = 1500 nM T18876 C6SGH7 9954562 Ki = 1300 nM T18876 C4UK2Q 9955802 Ki = 5.5 nM T18876 C6ZM4U 9959673 Ki = 4700 nM T18876 CCD30P 9960839 Ki > 100000 nM T18876 C4Z7BL 9965922 Ki = 1600 nM T18876 C5AF0B 9975502 EC50 = 15 nM T18876 CV67PS 10000048 EC50 = 34 nM T18876 CGP90V 10002871 EC50 = 1730 nM T18876 CHR8C2 10003118 EC50 = 44 nM T18876 CCD24K 10007859 IC50 = 158.49 nM T18876 CQ3GW6 10047541 IC50 > 10000 nM T18876 CH79JK 10069539 EC50 = 290 nM T18876 CQT1G4 10089562 EC50 = 21 nM T18876 CNE21V 10095268 Ki = 6309.57 nM T18876 COR8X7 10109445 Ki = 6.9 nM T18876 C6UI2Z 10111602 Ki = 610 nM T18876 CBYV78 10112486 Ki = 1100 nM T18876 C93DSI 10113454 Ki = 16 nM T18876 C4WVN0 10113722 EC50 = 39.81 nM T18876 C26QRM 10118889 Ki = 1000 nM T18876 CGF7K0 10120328 Ki = 0.31 nM T18876 C6BOW4 10144273 Ki = 19000 nM T18876 CBJ1G3 10145097 Ki = 2.4 nM T18876 CG4YV6 10157810 Ki = 6313 nM T18876 C6W9IC 10158725 Ki = 650 nM T18876 C4VN9H 10159697 Ki = 7 nM T18876 CM3SE6 10168694 Ki = 7100 nM T18876 C71GVU 10178073 Ki = 1900 nM T18876 CPF8H0 10181299 EC50 = 125.89 nM T18876 CEM21G 10181606 Ki = 3700 nM T18876 CS83AF 10189261 Ki = 0.37 nM T18876 C6X5CP 10202765 Ki = 1.6 nM T18876 CMD93W 10204257 Ki = 57 nM T18876 C4DLP9 10205205 Ki = 59 nM T18876 C78MPA 10208065 EC50 > 1000 nM T18876 CNT8H9 10221497 Ki = 68 nM T18876 CX32UD 10223809 EC50 = 25.12 nM T18876 CP8KN7 10227492 Ki = 1100 nM T18876 CZP7B5 10229201 Ki = 27 nM T18876 CFWB04 10247632 Ki = 443 nM T18876 C0ED9Y 10251023 IC50 > 10000 nM T18876 C81HOQ 10268898 EC50 = 2100 nM T18876 C47IJF 10269242 EC50 = 277 nM T18876 CQ0R3G 10270893 Ki = 2000 nM T18876 C89CXB 10271490 Ki = 2900 nM T18876 CZ21EM 10272306 Ki = 36 nM T18876 C8FH6E 10276417 EC50 = 199.53 nM T18876 CL7YG3 10287121 Ki = 2100 nM T18876 C40QFO 10291963 EC50 = 0.02 nM T18876 CK7M3E 10295421 EC50 = 0.2 nM T18876 C2J0PF 10298293 EC50 = 0.2 nM T18876 CV9QL7 10302378 Ki = 1100 nM T18876 C3C5IM 10322469 EC50 = 0.8 nM T18876 CB19MW 10402929 Ki = 10000 nM T18876 C0M2HU 10427236 Ki = 90 nM T18876 CT8UC2 10448293 EC50 = 4 nM T18876 C8ZB6N 10452108 EC50 = 0.5 nM T18876 CZ1XW6 10483360 Ki = 44000 nM T18876 CI5HA0 10648334 IC50 > 10000 nM T18876 C9YQG5 10670992 IC50 > 10000 nM T18876 C7GY6X 10739351 IC50 > 10000 nM T18876 CY8IB2 10740699 IC50 > 10000 nM T18876 C12SBH 10741017 IC50 > 10000 nM T18876 CG17HE 10741197 IC50 > 10000 nM T18876 CKST02 11122314 IC50 > 10000 nM T18876 CEI08Z 11155228 Ki = 620 nM T18876 CC8PQ2 11156167 EC50 = 8390 nM T18876 CF6EO3 11210487 Ki = 2800 nM T18876 C4S5MX 11249458 Ki = 0.91 nM T18876 CH98QW 11255960 Ki = 530 nM T18876 C70ESM 11269563 Ki > 20000 nM T18876 COS4C2 11294085 EC50 = 195 nM T18876 C9E4SW 11294166 Ki > 2900 nM T18876 CVD58I 11295611 Ki = 8.4 nM T18876 CIM8K7 11328569 EC50 = 705 nM T18876 CU5BA9 11337781 Ki = 900 nM T18876 CQU62G 11337782 Ki = 18 nM T18876 C4IK7Y 11339240 Ki = 0.7 nM T18876 CBP71Y 11362836 EC50 = 1220 nM T18876 CN2TG7 11387144 Ki = 0.68 nM T18876 C2KI7L 11398562 Ki = 240 nM T18876 CUWE27 11405770 Ki = 17 nM T18876 CXPO04 11408533 Ki > 20000 nM T18876 CP4LS0 11440167 EC50 = 0.2 nM T18876 CZ4K0P 11476788 Ki > 16500 nM T18876 CE2JA4 11488860 Ki = 6610 nM T18876 CW3YO5 11494768 IC50 > 10000 nM T18876 C94TIW 11502889 IC50 = 5.02 nM T18876 CHBR87 11502930 IC50 < 50 nM T18876 CQ6IU7 11509269 IC50 > 10000 nM T18876 CS2LR0 11516353 IC50 > 10000 nM T18876 CF2OM8 11539410 IC50 > 10000 nM T18876 CM7HK0 11551847 IC50 > 10000 nM T18876 C8Z5QJ 11561083 IC50 < 50 nM T18876 CJ2OE0 11575201 IC50 = 8.76 nM T18876 C1W2ZK 11577792 Ki = 0.97 nM T18876 C8HMG9 11582853 IC50 < 50 nM T18876 C7Y6XJ 11597294 Ki = 4400 nM T18876 C2M8HZ 11610353 IC50 > 10000 nM T18876 CGS72I 11618662 IC50 = 13.4 nM T18876 C9Y5ZT 11626153 IC50 = 94.3 nM T18876 C9L5VD 11631813 IC50 > 10000 nM T18876 CD7R5P 11631965 IC50 > 10000 nM T18876 CMB6F9 11653874 IC50 > 10000 nM T18876 C51UDK 11667741 IC50 > 10000 nM T18876 CAL96X 11683088 IC50 = 9.68 nM T18876 CW8RY9 11689895 IC50 > 10000 nM T18876 C9CM2R 11695689 IC50 > 10000 nM T18876 C3BSV4 11696697 Ki = 12 nM T18876 C97CZX 11697738 IC50 < 50 nM T18876 C8G3US 11718930 IC50 = 41.1 nM T18876 CF3XD2 11742697 EC50 = 44 nM T18876 CNYK74 11743212 Ki = 300 nM T18876 CGR4K8 11755846 EC50 = 6.1 nM T18876 CMB78A 11957776 Ki = 0.43 nM T18876 CR82PA 12112238 Ki = 1700 nM T18876 CX0M2W 12112239 Ki = 1100 nM T18876 C32GBT 12137443 EC50 = 0.04 nM T18876 CT34LO 13230981 Ki = 6 nM T18876 CO19GA 14372497 Ki > 2900 nM T18876 C06OGJ 15486805 IC50 > 10000 nM T18876 C0L3VU 15486806 IC50 > 10000 nM T18876 CU5J6N 15491229 Ki > 100000 nM T18876 CMG0Z1 15491230 Ki > 100000 nM T18876 CWQ8B9 15551228 Ki = 8000 nM T18876 CZ87CN 15907747 Ki = 3000 nM T18876 CVEO28 15907748 Ki = 6900 nM T18876 CLOY50 15947337 Ki = 0.28 nM T18876 C5AEZ8 15947448 Ki = 0.38 nM T18876 C6RZ4I 15947546 Ki = 0.27 nM T18876 CG2I7L 15947639 Ki = 0.95 nM T18876 C5UH1D 15947640 Ki = 0.32 nM T18876 CW46RS 15947856 Ki = 0.54 nM T18876 CIS83K 15947857 Ki = 0.79 nM T18876 C3L0RK 15948325 Ki = 0.74 nM T18876 CU21ID 15948329 Ki = 0.76 nM T18876 C94KAP 15948439 Ki = 0.48 nM T18876 CU8Q7F 15948440 Ki = 9.8 nM T18876 CZ7Q8L 15948441 Ki = 2.8 nM T18876 CV97OJ 15948442 Ki = 2.4 nM T18876 CDB13U 15948554 Ki = 0.27 nM T18876 CI41OM 15948558 Ki = 0.21 nM T18876 C8Q4NA 15948674 Ki = 3.3 nM T18876 CRBI38 15948788 Ki = 0.55 nM T18876 CIW0B8 15948789 Ki = 0.36 nM T18876 CRT3I2 15979081 EC50 = 91 nM T18876 CK4FJ8 16664733 IC50 = 24000 nM T18876 CI61TE 16678098 EC50 = 6.31 nM T18876 C14XYI 17747304 EC50 = 79.43 nM T18876 CRH47L 18444538 Ki = 80 nM T18876 C9PVK2 18444545 Ki = 3800 nM T18876 CT46SZ 18444548 Ki = 1600 nM T18876 CE4BP6 18444550 Ki = 2800 nM T18876 CN36PY 18444554 Ki = 740 nM T18876 C75GWD 18444556 Ki = 1300 nM T18876 C3E1JM 18444557 Ki = 150 nM T18876 C09BLO 18444558 Ki = 600 nM T18876 CHL9W5 18444559 Ki = 1000 nM T18876 C0OF3M 18444560 Ki = 1500 nM T18876 C5AZ0M 18444567 Ki = 20 nM T18876 CTDM65 18444572 Ki = 3000 nM T18876 CRK69M 18444582 Ki = 100 nM T18876 C9J3FX 18444585 Ki = 3000 nM T18876 C9UCJ8 18444587 Ki = 80 nM T18876 CK9X2G 18444588 Ki = 1300 nM T18876 C7JC6P 18444589 Ki = 2000 nM T18876 CG4W6T 18444596 Ki = 11 nM T18876 C8F7LD 18444607 Ki = 2400 nM T18876 C8JF2Q 18444611 Ki = 85 nM T18876 CQGL16 18444613 Ki = 3 nM T18876 CQK2D0 18444614 Ki = 22 nM T18876 CWC2K4 18444616 Ki = 20 nM T18876 CG5UO0 18444619 Ki = 0.3 nM T18876 CC52IJ 18444622 Ki = 1.3 nM T18876 CPK91U 18444625 Ki = 21 nM T18876 CMEG91 18444626 Ki = 5 nM T18876 CX7OT1 18444627 Ki = 3 nM T18876 C45YFP 18444628 Ki = 218 nM T18876 C4W1GT 18444629 Ki = 2 nM T18876 CID0R3 18444630 Ki = 14 nM T18876 CFM10U 18444632 Ki = 25 nM T18876 CH9JS0 18444679 Ki = 115 nM T18876 CS8M2G 18973764 Ki = 440 nM T18876 C49TJP 21079273 EC50 > 1000 nM T18876 C4T2IM 21079274 EC50 = 5.012 nM T18876 C6DFU2 21079275 EC50 = 5.012 nM T18876 C3UR0B 21079276 EC50 = 251.19 nM T18876 C1WC9R 21079279 EC50 > 1000 nM T18876 CBC79I 21079282 EC50 = 10 nM T18876 CH49UC 21079283 EC50 = 7.943 nM T18876 CI1WX4 21079296 EC50 = 199.53 nM T18876 CX08BC 21198692 Ki > 15000 nM T18876 CR37AJ 21362845 Ki = 28000 nM T18876 C6UT1I 21362849 Ki = 1200 nM T18876 C4IFY8 21362851 Ki = 1800 nM T18876 C9HQN0 21362853 Ki = 1000 nM T18876 C6F8QI 21362863 Ki = 21000 nM T18876 CL5O9E 21362867 Ki = 25000 nM T18876 C58NCB 21362869 Ki > 100000 nM T18876 CHS9L6 21362879 Ki = 760 nM T18876 CW7R1M 21362893 Ki = 1600 nM T18876 C9HD2W 21362900 Ki = 1100 nM T18876 CSUO46 21362905 Ki = 980 nM T18876 CJ65SZ 21362910 Ki = 2000 nM T18876 CFV24G 21362912 Ki = 700 nM T18876 C0UT6R 22008966 Ki = 1000 nM T18876 CJ4M7P 22008967 Ki = 1000 nM T18876 C9TSB7 22009003 Ki = 1000 nM T18876 C8SON3 22009004 Ki = 840 nM T18876 CAML12 22009006 Ki = 1500 nM T18876 C5DGQ4 22009008 Ki = 840 nM T18876 C5SJ2H 22009011 Ki = 930 nM T18876 C3D2LR 22990263 Ki > 10000 nM T18876 CF81SW 23582412 IC50 > 10000 nM T18876 CV4PX5 23634376 Ki = 0.44 nM T18876 CULW17 23654359 EC50 = 630 nM T18876 CO85UG 23660504 Ki = 1.5 nM T18876 C0AXU2 23660505 Ki = 7.5 nM T18876 CJW38X 23660675 Ki = 3.1 nM T18876 CFJL86 23660678 Ki = 0.33 nM T18876 CBU2S6 23660680 EC50 = 0.2 nM T18876 CD7KG8 23660841 Ki = 0.37 nM T18876 CJ2RC6 23660845 IC50 = 4.7 nM T18876 C8N1BM 23661014 Ki = 0.44 nM T18876 CP80HO 23661015 Ki = 1 nM T18876 CN4A2J 23661017 Ki = 30 nM T18876 CT07BI 23661189 Ki = 0.34 nM T18876 CP2S4J 23663736 Ki = 7200 nM T18876 CASU54 23696973 IC50 > 31622.78 nM T18876 CP72MI 24739203 EC50 = 3.981 nM T18876 C42LYP 24765153 Ki = 6549 nM T18876 CF72YI 24765671 Ki = 4.8 nM T18876 C31JZP 24765672 Ki = 2.7 nM T18876 C4QX7Y 24765675 Ki = 20.1 nM T18876 CF4EN6 24765766 Ki = 39.5 nM T18876 CL7Z9U 24765768 Ki = 0.81 nM T18876 CE1K3P 24765769 Ki = 56 nM T18876 CQ1F4V 24771582 EC50 = 280 nM T18876 C1ITO3 24771583 EC50 = 21000 nM T18876 CB2C4U 24944538 Ki = 0.48 nM T18876 CR6EM2 24944617 EC50 = 50.12 nM T18876 CKL5U3 24945854 EC50 = 19.95 nM T18876 CFQA40 24952577 Ki = 6.4 nM T18876 CD98IN 24952580 Ki = 1.3 nM T18876 C81WVN 24952927 Ki = 1.4 nM T18876 CZT83E 24952928 Ki = 0.63 nM T18876 C8YHX3 24953283 Ki = 0.87 nM T18876 CZ93FO 24953285 Ki = 0.72 nM T18876 C17JTY 24953286 Ki = 3.1 nM T18876 CFT0W5 24953624 Ki = 0.75 nM T18876 C42VMD 24953625 Ki = 2.5 nM T18876 C7B2EW 24953628 Ki = 2.9 nM T18876 CXQJ67 25002382 Ki = 0.31 nM T18876 CN5SH9 25003075 Ki = 0.23 nM T18876 C8TM3K 25015836 Ki = 1.2 nM T18876 CR38LC 25016088 Ki = 0.39 nM T18876 CD9NF6 25018911 Ki = 0.3 nM T18876 C1AJ7P 25019183 Ki = 0.16 nM T18876 C16NOI 25019184 Ki = 0.23 nM T18876 C6V3YF 25019185 Ki = 0.17 nM T18876 C3ZJ2T 25019433 Ki = 0.49 nM T18876 CC2WJ7 25019434 Ki = 0.34 nM T18876 CJ63ES 25019435 Ki = 0.52 nM T18876 CF29BG 25019694 Ki = 0.4 nM T18876 CUW16F 25019695 Ki = 0.4 nM T18876 C1CIE6 25019696 Ki = 0.48 nM T18876 C2CNM6 25019697 Ki = 0.66 nM T18876 C4J2BS 25195248 IC50 = 6200 nM T18876 CR10FW 30897313 IC50 = 3500 nM T18876 CNOF71 44138108 Ki > 11300 nM T18876 CSRV98 44157014 IC50 = 12500 nM T18876 C2AV1K 44190762 IC50 = 3700 nM T18876 C2O0NL 44230575 IC50 = 5480 nM T18876 CQ13MH 44234032 Ki = 1200 nM T18876 CR68BA 44250281 Ki > 10000 nM T18876 CN90FE 44269464 Ki = 1110 nM T18876 C1L0ET 44269468 Ki = 243 nM T18876 C5KRQ4 44269486 Ki = 28 nM T18876 CL6M2P 44269516 Ki = 35 nM T18876 CON8R9 44269520 Ki = 140 nM T18876 C6MBG0 44269521 Ki = 13 nM T18876 CZ3Q1L 44269523 Ki = 3.6 nM T18876 CRL61O 44269532 Ki = 66 nM T18876 C1Z4LU 44269540 Ki = 443 nM T18876 CM72FA 44269542 Ki = 1410 nM T18876 CN0JV2 44269543 Ki = 3500 nM T18876 C28UJH 44269544 Ki = 2.6 nM T18876 CR1IY6 44269568 Ki = 62 nM T18876 CI3C9O 44269596 Ki = 102 nM T18876 CC0EW9 44269597 Ki = 230 nM T18876 CY37TX 44289792 EC50 = 17 nM T18876 C6JAE2 44289921 Ki = 7.5 nM T18876 CDJV85 44289968 Ki = 7.4 nM T18876 CG8KT3 44289969 Ki = 2300 nM T18876 C68XKV 44289977 Ki = 140 nM T18876 CV7RO5 44289980 EC50 = 6100 nM T18876 C1H8MK 44290245 EC50 > 100000 nM T18876 CHZ21Q 44290257 Ki = 4.9 nM T18876 CO31WZ 44290262 EC50 = 50 nM T18876 COF9C2 44290263 Ki = 8.2 nM T18876 C4SEW6 44290266 Ki = 0.8 nM T18876 CEVM85 44290267 Ki = 4.2 nM T18876 C7RDN9 44290271 EC50 = 170 nM T18876 CN5RG9 44290272 Ki = 6.2 nM T18876 CZ59QY 44290312 EC50 = 360 nM T18876 CAV76T 44290314 Ki = 10 nM T18876 CJ59WE 44290315 EC50 > 10000 nM T18876 C8RA9P 44290316 EC50 = 42000 nM T18876 C4F8YR 44290494 Ki = 32 nM T18876 CS7RH0 44320126 Ki = 730 nM T18876 CLR9F5 44320272 Ki = 850 nM T18876 CKYS39 44320294 Ki = 1100 nM T18876 CH6TK1 44320321 Ki = 1000 nM T18876 CYI1O0 44320373 Ki = 4400 nM T18876 C0V3OA 44320388 Ki = 2900 nM T18876 C01HGT 44320405 Ki = 690 nM T18876 CS58ZQ 44320433 Ki = 1500 nM T18876 CS52ZR 44324368 Ki = 19000 nM T18876 CM72WE 44349503 Ki = 1700 nM T18876 C9PO1Q 44349528 Ki = 1100 nM T18876 C1R7HU 44349531 Ki = 1100 nM T18876 CHO7X0 44349551 Ki = 460 nM T18876 CLN63A 44377464 Ki > 40000 nM T18876 CJIS72 44390782 Ki = 4300 nM T18876 C43VIA 44390806 Ki = 1700 nM T18876 CB8H4V 44390831 Ki = 2400 nM T18876 CRFL02 44400189 Ki = 50 nM T18876 C68IYQ 44400223 Ki = 80 nM T18876 CR81DJ 44400307 EC50 = 110 nM T18876 CZK3R9 44400318 EC50 = 260 nM T18876 CWL1X4 44400355 Ki = 43 nM T18876 C76QVA 44402710 Ki > 10000 nM T18876 CRAX23 44402824 Ki > 10000 nM T18876 CIB2W5 44419347 Ki = 620 nM T18876 CF35LY 44419350 Ki = 440 nM T18876 CNK1X9 44419351 Ki = 1000 nM T18876 C91JXT 44419374 Ki = 2000 nM T18876 CNF4W2 44419379 Ki = 2000 nM T18876 CS3IW4 44419380 Ki = 960 nM T18876 CBQ01L 44419384 Ki = 960 nM T18876 CGS0P7 44442327 EC50 = 0.002 nM T18876 CF32IP 44442331 EC50 = 0.1 nM T18876 CZVA37 44442332 EC50 = 2 nM T18876 C0IV9J 44442334 EC50 = 3 nM T18876 C7HFG3 44442337 Ki = 117 nM T18876 CCV69D 44444714 Ki = 6000 nM T18876 CVH1E4 44444715 Ki = 330 nM T18876 CZ27AC 44444716 Ki = 44 nM T18876 CQL04T 44444719 Ki = 134 nM T18876 CE5MU6 44444720 EC50 = 0.1 nM T18876 CXQ5K3 44444721 Ki = 26 nM T18876 CW60FE 44444722 Ki > 50000 nM T18876 CDBE16 44450497 Ki > 16061 nM T18876 CE0ID1 44453376 Ki = 0.25 nM T18876 CT09SX 44453545 Ki = 0.43 nM T18876 C43AOW 44453566 Ki = 0.12 nM T18876 CV3M0X 44453572 Ki = 4.2 nM T18876 C6NRL2 44453656 Ki = 0.38 nM T18876 C1LE6O 44453657 Ki = 2 nM T18876 CC0N4T 44453997 Ki = 7.9 nM T18876 CH2K9C 44454020 Ki = 1 nM T18876 C3O7LT 44454021 Ki = 0.43 nM T18876 CV8IX1 44455046 Ki = 0.02 nM T18876 CRZ5K2 44455084 EC50 = 0.3 nM T18876 CD6B3W 44455115 EC50 = 3 nM T18876 CCY63H 44455157 Ki = 490 nM T18876 C3DQ5V 44455158 Ki = 27 nM T18876 C1CB7O 44455236 Ki = 1 nM T18876 CUHD74 44564571 IC50 = 20400 nM T18876 CA05LN 44564804 IC50 = 14600 nM T18876 C6XE0K 44564841 IC50 > 10000 nM T18876 CND54C 44564892 IC50 = 13000 nM T18876 C2VR6S 44564893 IC50 > 10000 nM T18876 C18GXI 44564937 IC50 > 10000 nM T18876 CZ74GB 44564990 IC50 = 10000 nM T18876 C0NF1S 44565193 IC50 > 10000 nM T18876 C07ODW 44570000 IC50 = 6498 nM T18876 CJKA53 44570666 IC50 = 7700 nM T18876 CSW92V 44570668 IC50 = 20800 nM T18876 CTW6L7 44570712 IC50 = 20800 nM T18876 CXQI89 44571354 IC50 = 7500 nM T18876 C5PT0Z 44626877 IC50 = 8178 nM T18876 CQIK27 44627395 IC50 = 10172 nM T18876 C4W1ZG 44627515 IC50 = 3647 nM T18876 C5AY6M 46220498 Ki > 2700 nM T18876 CS4F0X 46879894 IC50 = 18600 nM T18876 C2FR7X 46885690 IC50 = 15100 nM T18876 CN8D5V 46885691 IC50 = 2300 nM T18876 C9RP0X 46885735 IC50 = 8700 nM T18876 C0A2CI 46890616 Ki = 2.4 nM T18876 CW52VH 46890658 Ki = 0.38 nM T18876 CXQ2W0 46890659 Ki = 0.62 nM T18876 CQ20RC 46890660 Ki = 0.44 nM T18876 CTR7Q0 49850345 IC50 > 50118.72 nM T18876 CM06FG 50898361 Ki = 0.54 nM T18876 CF1ZU9 52945294 Ki = 610 nM T18876 C4K6BH 52946883 Ki > 10000 nM T18876 C7PSX2 53316600 Ki = 0.2 nM T18876 CIG1X0 53316601 Ki = 3 nM T18876 C73JVA 53317328 Ki = 1.8 nM T18876 C1RYL7 53317329 Ki = 2.3 nM T18876 CQ60OF 53317509 Ki = 0.28 nM T18876 C24RMK 53317842 Ki = 0.87 nM T18876 CKXW30 53317904 Ki = 0.97 nM T18876 CFS70H 53317905 Ki = 0.59 nM T18876 CV35WS 53318618 Ki = 76 nM T18876 CF5YO6 53319154 Ki = 0.32 nM T18876 CW15UJ 53319233 Ki = 0.44 nM T18876 CED3N4 53319234 Ki = 0.5 nM T18876 C02KNP 53320541 Ki = 0.33 nM T18876 C0O5ZH 53320542 Ki = 0.53 nM T18876 CL2D3H 53320543 Ki = 0.77 nM T18876 C5AJ1X 53320544 Ki = 2.3 nM T18876 C7S0AQ 53320545 Ki = 1.6 nM T18876 CWGA19 53321772 Ki = 0.67 nM T18876 C1BUP5 53321854 Ki = 1.9 nM T18876 C7RZ9E 53321855 Ki = 0.55 nM T18876 CK12ZF 53322687 Ki = 22 nM T18876 C2K9AV 53322911 Ki = 14 nM T18876 COCL81 53323010 Ki = 0.41 nM T18876 C5K3PJ 53323050 Ki = 0.37 nM T18876 C7CE5V 53323098 Ki = 0.11 nM T18876 C58KTH 53323099 Ki = 0.2 nM T18876 C3M2XH 53323176 Ki = 10 nM T18876 CE4MC5 53323177 Ki = 0.42 nM T18876 CV86GF 53323178 Ki = 3.8 nM T18876 CZ9M6V 53323903 Ki = 54 nM T18876 CI7N6P 53323904 Ki = 0.78 nM T18876 CW4SK1 53324453 Ki = 0.71 nM T18876 CVG7K3 53324525 Ki = 14 nM T18876 C95HQS 53325181 Ki = 30 nM T18876 CQWP93 53325182 Ki = 0.4 nM T18876 CWE36A 53325585 Ki = 0.34 nM T18876 C52QXE 53325764 Ki = 0.18 nM T18876 CJV90D 53325765 Ki = 0.16 nM T18876 C45YLC 53325766 Ki = 4.4 nM T18876 CJ5CM9 53325767 Ki = 0.32 nM T18876 C43OKB 53325840 Ki = 0.4 nM T18876 CT39HS 53325841 Ki = 29 nM T18876 C81KDF 53325842 Ki = 0.98 nM T18876 CVSF07 53326475 Ki = 0.66 nM T18876 CBK08J 53326912 Ki = 1.1 nM T18876 CWR1Z7 56665984 Ki = 2.5 nM T18876 CA1DF5 57392712 IC50 = 2 nM T18876 C96FQZ 57395059 EC50 = 0.5 nM T18876 C8RS3N 57396195 IC50 = 1000 nM T18876 CRUJ96 57399661 IC50 = 34 nM T18876 CVLQ48 57401413 IC50 = 42 nM T18876 C5JE1H 58824161 Ki = 1.3 nM T18876 C9U0ON 58824188 Ki = 3.6 nM T18876 CHA4Z3 58824190 Ki = 0.6 nM T18876 C8CO1U 58824194 Ki = 15 nM T18876 C87ZCR 58824196 Ki = 5 nM T18876 CUR1N2 58824201 Ki = 13 nM T18876 CC0YM5 58824204 Ki = 24 nM T18876 CV15PD 58905312 IC50 = 340 nM T18876 CFN2G3 58905313 IC50 = 181 nM T18876 CC30NM 58905340 IC50 = 400 nM T18876 C0H7KO 58905345 IC50 = 28.7 nM T18876 CP7A2U 58905349 IC50 = 37.9 nM T18876 CB1N8J 58905358 Ki = 73 nM T18876 C0EHD5 58905363 IC50 = 137 nM T18876 C7Z0CY 58905368 IC50 = 21.6 nM T18876 C6XTB8 58905379 IC50 = 545 nM T18876 C1CFM4 58905388 IC50 = 124 nM T18876 C0U1HA 59179260 Ki > 2700 nM T18876 CK7T6D 59179887 Ki > 2700 nM T18876 C4CIH9 59179917 Ki > 2700 nM T18876 CVC72I 59554822 EC50 = 73 nM T18876 CCXA68 59554824 EC50 = 320 nM T18876 C2EVC3 59554827 EC50 = 4.2 nM T18876 CNUA34 66857670 EC50 = 240 nM T18876 C1WA3L 66857738 EC50 = 4710 nM T18876 C1C3AF 66857975 EC50 > 10000 nM T18876 CUIV04 66857988 EC50 = 3380 nM T18876 CB56OD 66858036 EC50 > 10000 nM T18876 CU5V8I 66858111 EC50 = 465 nM T18876 CB2J4V 66978356 EC50 = 146 nM T18876 C4FHO2 67082722 EC50 = 2540 nM T18876 CGQA79 67082748 EC50 = 127 nM T18876 CVM9Q1 68503758 IC50 > 10000 nM T18876 CA15ND 68505312 IC50 > 10000 nM T18876 C0US2T 68505327 IC50 > 10000 nM T18876 CX8W7F 68508048 IC50 > 10000 nM T18876 C5NZO0 68747479 EC50 > 10000 nM T18876 C8H2JG 69147154 Ki = 1200 nM T18876 CJ7AY6 69753740 EC50 = 4600 nM T18876 C01YOJ 71452690 Ki = 2600 nM T18876 CQ5E0J 71455094 Ki = 9448 nM T18876 COK0V6 71458757 Ki = 902 nM T18876 C74PUE 71462285 Ki = 3183 nM T18876 C8XJ0I 71733818 IC50 > 10000 nM T18876 CXC78L 71733909 IC50 > 10000 nM T18876 C7B5XE 71733910 IC50 > 10000 nM T18876 CQ21ZD 71733911 IC50 > 10000 nM T18876 CZG0S2 71733912 IC50 > 10000 nM T18876 C4G2UR 72695027 IC50 = 5.62 nM T18876 CDFO42 72695136 Ki = 58 nM T18876 CX6T7A 72706947 EC50 = 0.476 nM T18876 C6PLC5 72722131 EC50 = 0.088 nM T18876 CU39ZO 72950089 EC50 = 0.021 nM T18876 CT7UE8 74762651 IC50 = 4.7 nM T18876 C80URK 76281184 IC50 = 82.5 nM T18876 C5M9TI 76281455 IC50 = 18 nM T18876 CYV9T6 76281721 IC50 = 23.8 nM T18876 CE5PC7 76281723 IC50 = 14.7 nM T18876 CN8ZJ3 76281993 IC50 = 286 nM T18876 CO7NW1 76282475 IC50 = 33.8 nM T18876 CR5VJ6 76282476 IC50 = 34.2 nM T18876 CB7C1F 76283442 IC50 = 134.2 nM T18876 C2AD8W 76283950 IC50 = 733.3 nM T18876 CZE4Y6 76283951 IC50 = 165.5 nM T18876 CB4YF5 76284214 IC50 = 12.8 nM T18876 CHM87Q 76284215 IC50 = 157.7 nM T18876 C56UWT 76284477 IC50 = 6.8 nM T18876 C70OMJ 78319379 IC50 = 0.28 nM T18876 CK6U1S 86707344 IC50 = 19.5 nM T18876 CKBM98 86707347 IC50 = 16.5 nM T18876 CCW04E 86707350 IC50 = 14.2 nM T18876 C2RB5X 86707352 IC50 = 39.8 nM T18876 C7NTM0 86707355 IC50 = 87.9 nM T18876 CU1N9D 86707358 IC50 = 84 nM T18876 CN0W2G 86707359 IC50 = 96.7 nM T18876 C9B7MN 86707361 IC50 = 1.61 nM T18876 C2O0YD 89914445 IC50 = 14.4 nM T18876 CBK49T 89914524 IC50 = 5.42 nM T18876 CT26QR 89914526 IC50 = 2.87 nM T18876 CY36MK 89914844 Ki = 126 nM T18876 CDL38B 89914863 Ki = 372 nM T18876 C6B2GO 90202290 IC50 = 7 nM T18876 CTC7L8 90202404 IC50 = 24.7 nM T18876 CL5NF3 90202434 IC50 = 5.2 nM T18876 C4EWG5 90202545 IC50 = 34.6 nM T18876 CX0DS7 90202554 IC50 = 43.7 nM T18876 CHS94I 90202558 IC50 = 15.3 nM T18876 C98WTC 90202587 IC50 = 4.3 nM T18876 CQ53MY 90202594 IC50 = 51.5 nM T18876 CDC26L 90202660 IC50 = 4.4 nM T18876 C5X6WK 90202705 IC50 = 63 nM T18876 CJCS45 90202707 IC50 = 257.1 nM T18876 CW98RM 90202708 IC50 = 22.1 nM T18876 CTQ07Y 90202748 IC50 = 611.7 nM T18876 C96YNT 90656140 Ki > 30000 nM T18876 CSL02I 90656141 Ki = 1400 nM T18876 CG84PK 90656142 Ki = 10000 nM T18876 C1L4YN 90656143 Ki > 10000 nM T18876 CRX83Z 90656144 Ki > 10000 nM T18876 CA0U4M 90656145 Ki > 10000 nM T18876 CT8CD9 90656146 Ki > 10000 nM T18876 C5DRA1 90656147 Ki > 10000 nM T18876 CZ7DL9 90656148 Ki > 10000 nM T18876 C1T5HW 90656149 Ki > 10000 nM T18876 C2K3TB 90656150 Ki > 10000 nM T18876 C62JZK 90656151 IC50 = 1200 nM T18876 CGN40X 90656152 IC50 = 10000 nM T18876 CWTO83 91810751 IC50 = 2.36 nM T18876 C71DHP 118174952 IC50 = 11.2 nM T18876 CEF26M 118174960 IC50 = 1.56 nM T18876 CQ8U9N 118174968 IC50 = 3.08 nM T18876 CR4DE7 118175009 Ki = 3.49 nM T18876 C6CG3R 118175029 IC50 = 4.49 nM T18876 C8JG5H 118190908 IC50 = 59.5 nM T18876 CD37EG 118190924 IC50 = 0.73 nM T18876 CLGE69 118191077 IC50 = 1.11 nM T18876 CF08NP 118191080 Ki = 8.04 nM T18876 C1XPI5 118191081 IC50 = 5.65 nM T18876 CB4R7K 118191085 Ki = 17 nM T18876 C46GPN 118191092 IC50 = 0.67 nM T18876 COF6C8 118191093 IC50 = 1.94 nM T18876 C4SY8T 118191094 IC50 = 0.67 nM T18876 CNY9D1 118191104 Ki = 1.98 nM T18876 CSJ4A9 118352160 EC50 > 10000 nM T18876 CE6L8I 118352177 EC50 > 10000 nM T18876 C8PKA7 118352211 EC50 > 10000 nM T18876 CPS7M4 118352285 EC50 > 10000 nM T18876 C7Z3HU 122180289 IC50 = 3200 nM T18876 C2NG1J 122180295 IC50 = 18000 nM T18876 C8ZRJ0 126495398 EC50 > 10000 nM T18876 C8SRZ5 126495427 EC50 > 10000 nM T18876 CD72CT 126495432 EC50 > 10000 nM T18876 CN72WL 126495463 EC50 > 10000 nM T18876 CV1A6C 126495491 EC50 > 10000 nM T18876 CYP3E5 126495507 EC50 > 10000 nM T18876 C2N7XJ 127026652 EC50 = 745 nM T18876 CX9M6D 127029402 EC50 > 10000 nM T18876 CWXR72 127029417 Ki > 50000 nM T18876 CW1O4F 127029692 EC50 > 10000 nM T18876 C0UJ5N 127037150 EC50 = 3 nM T18876 CN7IQ9 127041464 Ki > 19200 nM T18876 CJAQ90 127047381 Ki > 50000 nM T18876 CBCQ64 127047601 Ki > 10000 nM T18876 CTR62O 127052613 EC50 = 33 nM T18876 CGZR45 127052614 EC50 = 1900 nM T18876 COVY75 127052615 EC50 > 10000 nM T18876 CWNS03 129161002 IC50 = 4.2 nM T18876 CW2U4L 136216100 IC50 = 6.1 nM T18876 CJ0AS7 137633712 IC50 = 1790 nM T18876 C57KYA 137633794 IC50 = 302 nM T18876 CMF58L 137637160 IC50 = 61.4 nM T18876 CTF8G5 137640686 IC50 = 60.4 nM T18876 C9LOM6 137641524 IC50 = 175 nM T18876 C26CJB 137643633 IC50 = 2940 nM T18876 CFT3Q0 137646517 IC50 = 1210 nM T18876 CFQ8I6 137648241 IC50 = 370 nM T18876 CG9XQ2 137649916 IC50 > 5000 nM T18876 CQ5B6C 137661981 IC50 = 93.5 nM T18876 CA8QC3 141730897 IC50 = 32 nM T18876 CG4N2I 141730898 IC50 > 10000 nM T18876 C2P9GV 141730900 IC50 = 1.3 nM T18876 CQ9AD0 141730904 IC50 = 49.1 nM T18876 C1Y7PO 141730908 IC50 = 161.3 nM T18876 CK6E7L 141730914 IC50 = 12.9 nM T18876 C7B5WG 141730916 IC50 = 3.1 nM T18876 CC2B6T 141730922 IC50 > 10000 nM T18876 C62DUY 141730923 IC50 = 45.6 nM T18876 CSXG54 145965248 EC50 > 10000 nM T18876 CIS1V8 145966519 EC50 > 10000 nM T18876 CPGL36 145970635 Ki = 199.53 nM T18876 C54SAN 145971909 EC50 = 26 nM T18876 CGV2E8 145977227 EC50 = 2636 nM T18876 CLVI73 145978309 EC50 = 578 nM T18876 CBN09F 145989275 Ki = 31.62 nM T18876 CDN70S 146014480 IC50 = 0.4 nM T18876 CK8L2Y 155514752 IC50 > 1000 nM T18876 CFQ75G 155515639 IC50 = 29.8 nM T18876 CJE63B 155516014 IC50 = 646.6 nM T18876 CJ7H4A 155516871 IC50 = 330.2 nM T18876 C1PN7M 155519679 IC50 = 147.5 nM T18876 CH8I3U 155520059 IC50 = 365.6 nM T18876 C5JGT1 155521209 IC50 = 224.8 nM T18876 CSA51B 155521594 IC50 = 1970 nM T18876 CZ10RG 155522808 IC50 = 27.9 nM T18876 CZ1WI0 155524344 IC50 > 10000 nM T18876 CTC43H 155524501 IC50 = 96.8 nM T18876 CUY37E 155524726 IC50 = 10.5 nM T18876 C3JG9H 155527097 IC50 > 10000 nM T18876 CFJC61 155528854 IC50 = 9.3 nM T18876 C04SLA 155529710 IC50 > 10000 nM T18876 C7UY3Q 155529786 IC50 = 8.5 nM T18876 CKQ85H 155530587 IC50 > 10000 nM T18876 CEW58P 155531552 IC50 = 65.1 nM T18876 CN1A7X 155533165 IC50 = 275.5 nM T18876 CY6WO2 155534871 IC50 > 10000 nM T18876 CR08CI 155539333 IC50 > 10000 nM T18876 CI3X9J 155541822 IC50 = 52.1 nM T18876 C95LVU 155542414 IC50 = 147.7 nM T18876 CYL96R 155544290 IC50 = 751.1 nM T18876 C9EH8X 155545601 IC50 > 10000 nM T18876 C8J4FW 155546443 IC50 = 17.4 nM T18876 CDC6V0 155548433 IC50 = 65.5 nM T18876 C5E3WI 155548550 IC50 > 10000 nM T18876 CG90YK 155549272 IC50 = 2315.7 nM T18876 CH0IO3 155550848 IC50 = 23 nM T18876 C4ZV6P 155552440 IC50 = 119.4 nM T18876 C2NI0O 155554096 IC50 = 13.9 nM T18876 C82RVN 155554217 IC50 = 4.6 nM T18876 C8P0OX 155555000 IC50 = 13.9 nM T18876 CXN9L5 155555513 IC50 = 118.8 nM T18876 C8SD3P 155555737 IC50 = 1422 nM T18876 CYF6N3 155556156 IC50 = 54.6 nM T18876 CU6YX3 155559165 IC50 = 68.8 nM T18876 CDN3M5 155559561 IC50 = 15.9 nM T18876 CG0TJ2 155559571 IC50 > 1000 nM T18876 C6WS0V 155560334 IC50 = 57.9 nM T18876 CT3GK1 155560972 IC50 > 10000 nM T18876 C8OEJ3 155561196 IC50 = 221.9 nM T18876 CZ62WJ 155563161 IC50 = 183 nM T18876 C74HWT 155564781 IC50 > 10000 nM T18876 CJ1E3W 155564876 IC50 > 10000 nM T18876 CC37GD 155565953 IC50 > 10000 nM T18876 C8OM1K 155566216 IC50 > 10000 nM T18876 C7QV0H 155568097 IC50 > 10000 nM T18876 CA5WB6 155568276 IC50 = 3118 nM T18876 C4VE9P 155568436 IC50 = 75.3 nM T18876 D02LXJ 9813912 Ki = 4400 nM T18876 D02MXT 24952929 Ki = 0.56 nM T18876 D02SAD 44419388 Ki = 6200 nM T18876 D03OYD 5311240 IC50 > 10000 nM T18876 D07JMB 44289922 EC50 = 0.065 nM T18876 D07UDT 15551229 Ki = 890 nM T18876 D08MNO 25886893 Ki > 10000 nM T18876 D08ZYC 11595431 Ki < 3162.28 nM T18876 D0H5TU 11524454 IC50 = 6.59 nM T18876 D0I0UI 5311232 Ki = 7 nM T18876 D0J9PG 119461 Ki > 100000 nM T18876 D0O9ES 5311053 IC50 > 10000 nM T18876 D0S2LO 9864831 Ki = 1.2 nM T18876 D0TA0L 23685469 Ki = 1020 nM T18876 D0Y1IF 23664784 Ki > 10000 nM T18876 D0Z3XJ 9817405 Ki = 3100 nM T16987 D00STL 644241 Ki = 302 nM T16987 D01MUR 68844 Ki = 3 nM T16987 D03QGM 5355 Ki = 3.9 nM T16987 D03RTS 2662 Ki = 18 nM T16987 D03UOT 785 Ki = 7800 nM T16987 D04AIT 5280445 Ki = 60.3 nM T16987 D05OFX 219078 Ki = 3713 nM T16987 D05UYW 5284549 Ki = 3 nM T16987 D07HBX 338 Ki = 8800 nM T16987 D07INV 3295 Ki = 22 nM T16987 D07MGA 72281 Ki = 454.1 nM T16987 D07VDZ 5284627 Ki = 3.8 nM T16987 D09NIA 2732 Ki = 4.5 nM T16987 D09VAZ 5565 Ki = 57000 nM T16987 D0AZ3C 5291 Ki = 980 nM T16987 D0AZ8C 5213 Ki = 9050 nM T16987 D0C2II 4100 Ki = 3.4 nM T16987 D0C8EU 5394 Ki > 50000 nM T16987 D0C8FX 3005837 Ki = 5400 nM T16987 D0E1SW 1986 Ki = 2.5 nM T16987 D0H8FH 3702 Ki = 10 nM T16987 D0J4GO 3038 Ki = 50 nM T16987 D0J7RK 36811 Ki = 4350 nM T16987 D0K0OZ 5702160 Ki = 45.3 nM T16987 D0K1QD 3998 Ki = 0.3 nM T16987 D0K8KX 5280343 Ki = 9390 nM T16987 D0L4JT 5333 Ki = 37 nM T16987 D0L6DA 119607 Ki = 13 nM T16987 D0L7FM 4911 Ki = 1245 nM T16987 D0OT0O 44561 Ki = 1290000 nM T16987 D0PQ3G 3440 Ki = 261 nM T16987 D0SH3I 387447 Ki = 5870 nM T16987 D0U5QK 1983 Ki = 4100 nM T16987 D0V8QT 2708 Ki > 50000 nM T16987 D0VM2L 68740 IC50 = 316 nM T16987 D0Y2IZ 5560 Ki = 312 nM T16987 D0Z3EI 6038 Ki = 93 nM T16987 D04IIU 216468 Ki = 3 nM T16987 D04PBH 5280804 Ki = 52.1 nM T16987 D05NJI 5287541 Ki = 12 nM T16987 D05ZXZ 491941 Ki = 77.2 nM T16987 D06DMQ 59472121 Ki > 50000 nM T16987 D08BXT 1102 Ki = 44100 nM T16987 D09XQU 135413511 Ki > 50000 nM T16987 D0I7MT 5281807 Ki = 515 nM T16987 D0L6HN 996 Ki = 9200 nM T16987 D0U3EP 445154 Ki = 950 nM T16987 D0V0UK 82267 Ki = 830000 nM T16987 D03SLR 445858 Ki = 9780 nM T16987 D0F8XZ 19890 Ki = 95200 nM T16987 D0NH9P 135 Ki = 4800 nM T16987 D07XPE 8249 Ki > 50000 nM T16987 D0LD9S 1103 Ki = 27600 nM T16987 CI0WH9 72 Ki = 4090 nM T16987 CU12QE 1203 Ki = 4720 nM T16987 C6O0MZ 1491 Ki = 7500 nM T16987 CO4X7B 2456 IC50 = 8442 nM T16987 C5L7VX 2871 Ki = 9520 nM T16987 CQ0D8J 3469 Ki = 7300 nM T16987 CJ2F6P 5056 Ki = 8130 nM T16987 CDJ4K6 5987 Ki = 700000 nM T16987 CUP2F4 7043 Ki = 8360 nM T16987 C1CVT7 7121 Ki = 6700 nM T16987 C6NC4O 7414 Ki = 2770 nM T16987 CJKY76 7420 Ki = 3530 nM T16987 C6QYD8 8434 Ki = 8600 nM T16987 CHP7I1 9016 Ki = 4020 nM T16987 CLYZ50 9338 Ki = 7200 nM T16987 CNM7L3 10199 Ki = 4.1 nM T16987 CBIR94 10313 Ki = 9510 nM T16987 CV5PC3 11568 Ki = 7700 nM T16987 CL80QG 11820 Ki = 83.5 nM T16987 CNI85U 15109 Ki = 8230 nM T16987 CQ4C5U 16523 Ki = 950 nM T16987 CNGB21 20098 Ki = 850 nM T16987 C3LA1Z 20161 Ki = 8500 nM T16987 CMK0O4 20825 Ki = 4.3 nM T16987 CG04AY 26518 Ki = 280 nM T16987 CDK20Z 27290 Ki > 50000 nM T16987 C69RDT 32204 Ki = 14600 nM T16987 C4OU6D 35703 Ki = 8200 nM T16987 CY2GU3 60582 Ki = 0.52 nM T16987 C5MJH8 64789 Ki = 2750 nM T16987 CN94KU 65008 Ki = 810 nM T16987 C1NQ8E 65188 Ki = 25700 nM T16987 CT6YO0 66548 Ki = 960 nM T16987 CMXS19 66814 Ki = 6 nM T16987 CJ1Z2R 67125 Ki = 950 nM T16987 C0ZK7U 67284 Ki = 7800 nM T16987 CWXE69 67756 Ki = 76.1 nM T16987 C26PTJ 67760 Ki = 135 nM T16987 CVI38F 69809 Ki = 690 nM T16987 CX4HM3 70653 IC50 = 8570 nM T16987 C8U0VH 72597 Ki = 0.78 nM T16987 CU79WI 74093 Ki = 176 nM T16987 CTMF08 75076 Ki = 840 nM T16987 C0I4UT 75077 Ki = 830 nM T16987 C7L1RO 75522 Ki = 7.9 nM T16987 CE5RZ1 76509 Ki = 520 nM T16987 C9V0ME 77547 Ki = 830 nM T16987 C6TS8J 77548 Ki = 750 nM T16987 CRXH06 77553 Ki = 7.8 nM T16987 CX47BZ 78479 Ki = 68000 nM T16987 CCK8E1 79611 Ki = 0.63 nM T16987 C5BFK4 87432 Ki = 730 nM T16987 CM72DQ 90631 Ki = 160 nM T16987 CB5R7Y 92229 Ki = 105 nM T16987 CB81UG 93577 Ki = 8.5 nM T16987 C2GI9X 95801 IC50 = 4280 nM T16987 C40RWH 95840 Ki = 94 nM T16987 C21JNS 95841 Ki = 18.7 nM T16987 CA9YN2 99477 Ki = 33.9 nM T16987 CV76MT 100187 Ki = 15600 nM T16987 CGM6A9 101263 Ki > 1000 nM T16987 CN19UT 129695 Ki = 190 nM T16987 CCK5Y6 133125 Ki = 3.2 nM T16987 CVB67D 134560 Ki = 85 nM T16987 CJ0FR9 155148 Ki = 8350 nM T16987 C50XVJ 159772 Ki = 480 nM T16987 C8AO0Z 165323 Ki = 36 nM T16987 CU3WG6 179620 Ki = 7440 nM T16987 CE1VJ6 191826 Ki = 53 nM T16987 C1N3AY 199210 Ki = 170 nM T16987 C2GHM7 202375 IC50 = 3302 nM T16987 CSMP84 219987 Ki = 9100 nM T16987 C9K3VU 220023 IC50 = 266 nM T16987 CEZU63 221227 Ki = 1170 nM T16987 C2ED9N 236541 Ki = 45.1 nM T16987 C14USE 239728 Ki = 710 nM T16987 CW1E5G 239730 Ki > 50000 nM T16987 C6D1LY 246499 Ki = 18.7 nM T16987 CLV79E 260228 Ki = 430 nM T16987 CU45WA 260244 Ki = 15600 nM T16987 C3QV5H 287064 Ki = 960 nM T16987 C26HNY 289493 Ki = 600 nM T16987 C83MLQ 295450 Ki = 2910 nM T16987 COE9A7 306924 Ki = 67.3 nM T16987 CAUO79 306968 Ki = 7.3 nM T16987 CM2N3X 307505 Ki = 8.5 nM T16987 C3W0AQ 307522 Ki = 61.2 nM T16987 C3WZI1 308397 Ki = 10.3 nM T16987 C6AKQ8 308411 Ki = 8.8 nM T16987 CL4GF1 308432 Ki = 7.5 nM T16987 C96DKW 310360 Ki = 4.5 nM T16987 CY13EN 311156 Ki = 7.6 nM T16987 C12PJC 313721 IC50 = 174 nM T16987 COI7H8 317746 Ki = 5.4 nM T16987 CG3J6Q 323350 Ki = 0.55 nM T16987 CTX0Z3 327169 Ki = 640 nM T16987 CXZ14S 341082 Ki = 13410 nM T16987 CP7X9H 342056 Ki > 10000 nM T16987 CMS5W4 343662 Ki = 36.5 nM T16987 CH1C9B 351361 Ki = 0.66 nM T16987 CM9V8O 388547 Ki = 4 nM T16987 CT3ZU4 388776 Ki = 10200 nM T16987 CH21KA 389641 Ki = 175000 nM T16987 C6CQO3 389642 Ki = 165000 nM T16987 CH0F9P 390929 Ki = 570 nM T16987 CNPZ40 394897 Ki = 2.8 nM T16987 C7HME8 439246 Ki = 44.3 nM T16987 CA8C5N 439514 Ki = 780 nM T16987 CC54LQ 450256 IC50 = 437 nM T16987 C5HM8E 474578 Ki = 53.1 nM T16987 CL0M9Y 482317 Ki = 880 nM T16987 CHF2Y9 493949 Ki = 766 nM T16987 C02DMG 504302 Ki = 46.5 nM T16987 CU7XE2 504303 Ki = 75.1 nM T16987 CNLT49 504304 Ki = 77 nM T16987 C49CNT 519869 Ki = 720 nM T16987 CJ7FR6 533728 Ki = 1105 nM T16987 C24ASH 539731 Ki = 7 nM T16987 C7EBA4 540544 Ki = 695.2 nM T16987 CFU6X9 560256 Ki = 798 nM T16987 CGHE12 607195 Ki = 76.5 nM T16987 CIK9S3 607305 Ki = 37.9 nM T16987 CP3SF2 609637 Ki = 48600 nM T16987 C1DX6J 640625 Ki = 96000 nM T16987 CH05FZ 648662 Ki = 517.7 nM T16987 C6PTC3 658040 Ki = 1780 nM T16987 CU9ZY6 670087 Ki = 72.4 nM T16987 CYGK68 676946 Ki = 490 nM T16987 C4YWI2 702292 Ki = 0.66 nM T16987 CYZ9O5 703304 Ki = 814.4 nM T16987 C9JH0M 706033 Ki = 440 nM T16987 C7ZE6K 706849 Ki = 2540 nM T16987 CK7DO5 708535 Ki = 39 nM T16987 CK9HY0 716763 Ki = 1.2 nM T16987 C8J4SO 724642 Ki = 83 nM T16987 C61NGE 724799 Ki = 35.5 nM T16987 C8G7EC 730672 Ki = 5.3 nM T16987 CNJZ35 738819 Ki = 50000 nM T16987 CV6Y7U 740560 IC50 = 179 nM T16987 CZM6W0 742873 Ki = 0.57 nM T16987 CLG6H5 746816 Ki = 0.98 nM T16987 CRIJ01 747569 Ki = 24 nM T16987 CW90GV 767467 Ki = 30.2 nM T16987 CV79DU 776418 Ki = 5500 nM T16987 CO1KN3 788171 Ki = 6.3 nM T16987 CA2B8X 792066 Ki = 9.4 nM T16987 CM0VX3 809685 Ki = 38.4 nM T16987 C6LN8S 816982 Ki = 2400 nM T16987 C5BGW9 818267 Ki > 50000 nM T16987 CJP5D4 818647 IC50 = 226 nM T16987 CVJZ57 818753 Ki = 41.9 nM T16987 CF93TC 821388 Ki = 770 nM T16987 C5VJZ0 822776 Ki = 0.64 nM T16987 CTD64N 834412 Ki = 427 nM T16987 C51FVL 906840 Ki = 9.4 nM T16987 CKV7B6 917551 Ki = 4.4 nM T16987 C4I3PJ 922062 Ki = 6.6 nM T16987 CRGQ70 927433 Ki = 910 nM T16987 CO7XW0 928228 Ki = 573.2 nM T16987 C6XQO2 940540 Ki = 38500 nM T16987 C4L9QD 943114 Ki = 48.9 nM T16987 COH62A 943115 Ki = 36.5 nM T16987 CX3U0S 975396 Ki > 50000 nM T16987 CZ3WK7 983751 Ki = 26.1 nM T16987 CN71CV 989611 Ki = 4.3 nM T16987 CJ2S0M 1070919 Ki = 8.9 nM T16987 CYS9A2 1070922 Ki = 0.6 nM T16987 CM2C5N 1070928 Ki = 2.3 nM T16987 COM2R4 1070933 Ki = 0.72 nM T16987 CDK1Z2 1085887 Ki > 50000 nM T16987 CA67JK 1124687 Ki = 1 nM T16987 C4QX1Z 1146666 Ki = 91.5 nM T16987 CJ82NF 1178394 Ki = 8.7 nM T16987 C7A8VI 1211699 Ki = 80.3 nM T16987 CYF34N 1211700 Ki = 0.9 nM T16987 C7QP5E 1213792 Ki = 4.9 nM T16987 C6T0NU 1230924 Ki = 18.5 nM T16987 C9IBF8 1241259 Ki = 6.8 nM T16987 CF1N3S 1277269 Ki > 50000 nM T16987 CL87AM 1286568 Ki = 10.4 nM T16987 CA1I9S 1286583 Ki = 38.5 nM T16987 CE6W7O 1287222 Ki = 446.6 nM T16987 CP60YD 1294363 Ki = 8.9 nM T16987 C5XNB4 1307068 Ki = 250 nM T16987 C40CKN 1316238 Ki = 27.3 nM T16987 CDWO53 1346695 Ki = 3.4 nM T16987 CC3G1N 1377410 Ki = 9.7 nM T16987 C9DY2L 1488548 Ki = 81500 nM T16987 CN5I0K 1505151 Ki = 28.4 nM T16987 CAHP42 1548275 Ki = 422 nM T16987 CORY25 1581900 Ki = 15.11 nM T16987 C40YCV 1655994 Ki = 61.6 nM T16987 CU7KR6 1738244 Ki = 34 nM T16987 C7XSO5 1748172 Ki = 72.5 nM T16987 CGKP07 1748225 Ki = 7.4 nM T16987 C98OLG 1775694 Ki = 9.1 nM T16987 CY20OQ 1945421 Ki = 0.65 nM T16987 CTF8R5 1957305 Ki = 47 nM T16987 C1DWG0 1989902 Ki = 6 nM T16987 CDQR23 2049187 Ki = 8.5 nM T16987 CSQJ97 2065546 Ki = 1841 nM T16987 CTK8C6 2089520 Ki = 150 nM T16987 C93VNU 2089779 Ki = 29 nM T16987 C3W4PG 2192287 Ki = 79 nM T16987 C2O9YS 2196398 Ki > 50000 nM T16987 CQS3A7 2207483 Ki = 56.6 nM T16987 CEW2Q3 2283723 Ki = 40 nM T16987 CGW6L4 2318645 Ki = 540 nM T16987 C1V0KL 2357187 Ki = 0.67 nM T16987 C3BJ4K 2368995 Ki = 46.8 nM T16987 CTJ42W 2368997 Ki = 3115 nM T16987 C4TD8M 2388085 Ki = 46.6 nM T16987 C1TW9F 2457081 Ki = 41 nM T16987 CJ10IX 2470552 Ki = 0.59 nM T16987 CR65UH 2471990 Ki = 2520 nM T16987 C95INQ 2476733 Ki = 4.6 nM T16987 C75SLD 2496330 Ki = 0.43 nM T16987 C2H4KT 2520594 Ki = 0.86 nM T16987 C8YH7W 2733779 Ki = 54 nM T16987 C0V7XB 2733782 Ki = 43 nM T16987 C0W8UL 2735045 Ki = 814 nM T16987 CQ70UR 2755708 Ki = 121 nM T16987 CU60ZB 2755709 Ki = 19.8 nM T16987 CNG69U 2755712 Ki > 50000 nM T16987 C58ISM 2755728 Ki = 3 nM T16987 CCOI52 2797418 Ki > 10000 nM T16987 CPO6W3 2813478 Ki = 2.3 nM T16987 CUI4Y8 2814914 Ki = 41 nM T16987 CLFB40 2815883 Ki = 8.1 nM T16987 CDSN81 2826269 Ki = 50.6 nM T16987 CBPO81 2882281 Ki = 18 nM T16987 CE2GR3 2900806 Ki = 21500 nM T16987 CW9M7A 2952488 Ki = 28.1 nM T16987 CFO90D 2952737 Ki = 2690 nM T16987 C61OTP 2991092 Ki = 49.9 nM T16987 CZEH20 3003616 Ki = 57.3 nM T16987 CJ9LZ7 3051101 Ki = 730 nM T16987 CN2Y5M 3083616 Ki = 7840 nM T16987 C9GT5Z 3083928 Ki = 18200 nM T16987 CQI7A2 3133127 Ki = 90 nM T16987 CXU4J8 3377675 Ki = 8 nM T16987 C1K6IA 3379075 Ki = 4.5 nM T16987 CIS69V 3440976 Ki = 9.4 nM T16987 CT1NB8 3441996 Ki = 3.2 nM T16987 CIXH89 3516083 Ki = 2.1 nM T16987 C0VI6O 3524248 Ki = 4500 nM T16987 CKTY04 3538605 Ki = 46.1 nM T16987 C86GSL 3542746 Ki = 4 nM T16987 CHGS79 3551941 Ki = 65.9 nM T16987 C9L1HS 3586494 Ki = 0.53 nM T16987 C4WZG2 3657160 Ki = 24.6 nM T16987 C3REH6 3703019 IC50 = 248 nM T16987 CQ5F9P 3724005 Ki = 13.6 nM T16987 C1JU9P 3774719 Ki = 7.1 nM T16987 C2SY4L 3856570 Ki > 10000 nM T16987 CI3KT8 3936209 Ki = 105 nM T16987 CV0KG3 3950536 Ki = 51.9 nM T16987 CJ6D2S 3970972 Ki = 0.57 nM T16987 C8DZ4B 4121769 Ki = 2.8 nM T16987 C9O0GV 4158561 Ki = 0.54 nM T16987 CT57HM 4204917 Ki = 6.8 nM T16987 CV6BJ7 4262171 Ki = 72.9 nM T16987 CUT26E 4274816 Ki > 50000 nM T16987 CUE97L 4276695 Ki = 70.7 nM T16987 CJ63TI 4578038 Ki = 0.94 nM T16987 CE5LO8 4578265 Ki = 43.9 nM T16987 C7RS2F 4583704 Ki = 1 nM T16987 CAPM27 4598704 Ki > 50000 nM T16987 CLSY09 4626049 Ki = 840 nM T16987 CPX3W6 4650747 Ki = 430 nM T16987 CTM71V 4654716 Ki = 428 nM T16987 CWXE71 4718084 Ki = 6.3 nM T16987 C6RC3L 4718087 Ki = 5.7 nM T16987 CRL7B4 4718142 Ki = 8.5 nM T16987 CJM5F3 4718971 Ki = 37.7 nM T16987 C6B0OY 4723880 Ki = 43.1 nM T16987 C0MFT8 4801151 Ki = 16 nM T16987 CSC7B8 4803242 Ki = 7.1 nM T16987 CUA65R 4857564 Ki = 92.7 nM T16987 CX8C3P 4961927 Ki = 7.7 nM T16987 CX3RJ9 5005133 Ki = 810 nM T16987 CIP6Q8 5017140 Ki = 92.7 nM T16987 C7JBU0 5019114 Ki > 50000 nM T16987 CF94ER 5032527 Ki = 17 nM T16987 C49FDN 5046067 Ki = 42.8 nM T16987 C4OAL9 5070078 Ki = 7500 nM T16987 CN31CX 5071527 Ki = 4.4 nM T16987 CU8E4B 5133468 Ki = 880 nM T16987 C89OCE 5155717 Ki = 0.62 nM T16987 CM9N8G 5161767 Ki = 9.3 nM T16987 C4HB1G 5172319 Ki = 2.8 nM T16987 CI8JY0 5172475 Ki = 4 nM T16987 CFQ62G 5232078 Ki = 1490 nM T16987 C4SV5T 5273568 Ki = 7450 nM T16987 CU4E5S 5273569 Ki = 7700 nM T16987 CZS0G5 5276565 IC50 > 10000 nM T16987 C3JN0F 5277465 IC50 > 10000 nM T16987 CRJK67 5277481 IC50 > 10000 nM T16987 CYF7S5 5277490 IC50 = 88 nM T16987 CD1LZ7 5278580 Ki = 4.9 nM T16987 CNZ73E 5280567 Ki = 8100 nM T16987 CN10FM 5281793 Ki = 39.8 nM T16987 CA18OQ 5316302 Ki = 9120 nM T16987 CTJ01E 5317485 Ki = 9100 nM T16987 CI58XK 5319562 Ki = 810 nM T16987 CNO53D 5321265 Ki = 790 nM T16987 CP0R5H 5336569 Ki = 402.2 nM T16987 C8PS4E 5358858 Ki = 700 nM T16987 CXEW32 5491996 Ki = 9070 nM T16987 C7RG3L 5496307 Ki = 7750 nM T16987 CX71JE 5682293 Ki = 6.5 nM T16987 CWYU91 5742696 Ki = 7940 nM T16987 CU0FW5 5743063 Ki = 7640 nM T16987 C4VZP8 5765787 Ki = 0.66 nM T16987 CWL5R2 5765789 Ki = 5.2 nM T16987 CK0M4A 5910585 Ki = 830 nM T16987 CHJ3V8 6102658 Ki = 370 nM T16987 CS4KQ6 6482974 Ki = 830 nM T16987 C9L8AX 6537802 Ki = 54 nM T16987 C65FRB 6852128 Ki = 1.5 nM T16987 CK85ZF 7022526 IC50 = 255 nM T16987 C0W5GD 7130726 Ki = 9.9 nM T16987 CWL9C2 7382212 Ki = 5.1 nM T16987 C75SBG 7382231 Ki = 2760 nM T16987 C6U9MT 7382238 Ki = 25.1 nM T16987 CY57CX 7382249 Ki = 15 nM T16987 CKCM96 7463376 Ki = 9310 nM T16987 CDCP43 7766335 Ki = 8890 nM T16987 C95AKP 7794397 Ki = 26 nM T16987 C1EKW8 7996519 Ki = 7.3 nM T16987 C67SFK 8084575 Ki = 21.1 nM T16987 CQ0Z4E 8098235 Ki = 14 nM T16987 CSW01Z 8272034 Ki = 3.9 nM T16987 C9BAM4 8281641 Ki = 0.59 nM T16987 C3WQ9M 8866559 Ki = 0.67 nM T16987 C5CS1Y 9314410 Ki = 50.5 nM T16987 C3SA2N 9314413 Ki = 96.2 nM T16987 C47VSJ 9572721 Ki > 10000 nM T16987 CIJ25V 9794947 IC50 = 5440 nM T16987 C7SRM4 9837496 IC50 = 5590 nM T16987 CY47OI 9998322 Ki = 4.5 nM T16987 CNKD31 10016330 Ki = 75.8 nM T16987 C4UEV9 10016475 Ki = 6.6 nM T16987 CF6RN0 10018880 Ki = 0.35 nM T16987 CX2W9O 10037048 IC50 = 6970 nM T16987 C5X7GY 10059582 Ki = 458.7 nM T16987 C69DPZ 10068042 IC50 = 855 nM T16987 CY8F0E 10076040 Ki = 8510 nM T16987 C0P5XV 10081897 Ki = 74.3 nM T16987 CD58EL 10083644 Ki = 29400 nM T16987 C7WU0A 10107532 Ki = 96.6 nM T16987 CXD91O 10136406 Ki = 91.9 nM T16987 CVRZ27 10198038 IC50 = 7260 nM T16987 CJV68L 10220266 Ki = 42.5 nM T16987 CQ8A0I 10328097 Ki = 399.7 nM T16987 CN40WD 10331524 Ki = 70.8 nM T16987 CUE81P 10337354 Ki = 4.7 nM T16987 C3HBY6 10375558 Ki = 55 nM T16987 CVIN94 10439991 Ki = 408.9 nM T16987 C6TYP0 10467861 Ki = 48.2 nM T16987 CD41CA 10512636 Ki = 783.8 nM T16987 C73KXU 10586607 Ki = 25600 nM T16987 C9TSQ6 10632698 Ki = 6200 nM T16987 CVHO36 10692638 Ki = 348 nM T16987 C6D2TJ 10712038 Ki = 1875 nM T16987 C2ZLE4 10737428 Ki = 52.9 nM T16987 C6EPH9 10919571 Ki = 6.8 nM T16987 C3WN6P 10931938 Ki = 685 nM T16987 C7FP4E 10932133 Ki = 3.4 nM T16987 CGI4X1 10933094 Ki = 8.4 nM T16987 CN27BY 10953838 Ki = 26500 nM T16987 CQBP46 11061197 Ki = 3 nM T16987 C8C6ER 11069133 Ki = 13 nM T16987 COGV98 11074431 Ki > 20000 nM T16987 CMK4Y0 11096006 Ki = 24.9 nM T16987 CWB10K 11103986 Ki = 4.8 nM T16987 CYQ01S 11115351 Ki = 3.9 nM T16987 CH6IE3 11117198 Ki = 7.7 nM T16987 C8X2DC 11127784 Ki = 3 nM T16987 C5WS3E 11147931 IC50 = 7270 nM T16987 CHC42Y 11245700 Ki = 13 nM T16987 CGE40M 11245996 Ki = 5.1 nM T16987 CCSA87 11280465 Ki = 90.2 nM T16987 CF15AS 11287957 Ki = 15.5 nM T16987 C3CDO1 11309586 Ki = 808 nM T16987 CRP08M 11310883 IC50 = 6640 nM T16987 CHA0V5 11321514 Ki = 860 nM T16987 CV80KU 11346010 Ki = 13900 nM T16987 C8PM3Z 11353795 Ki = 5 nM T16987 CM8Y1J 11367571 IC50 = 4650 nM T16987 CG1A5D 11427826 Ki = 1348 nM T16987 CUR65I 11441308 Ki = 18 nM T16987 CFER43 11467281 Ki = 7 nM T16987 CQ1D6E 11470070 IC50 = 7440 nM T16987 CU8YH7 11533895 Ki = 19 nM T16987 CIMD40 11578176 Ki = 8510 nM T16987 CDS25O 11593765 IC50 = 6000 nM T16987 C9QL2F 11615432 Ki = 181.5 nM T16987 C95PYS 11667431 Ki = 1.9 nM T16987 C9JR2I 11674590 Ki = 7420 nM T16987 CF8IT6 11696964 Ki = 3.3 nM T16987 CHAN30 11714982 Ki = 16 nM T16987 CH7Q5S 11777250 Ki = 8 nM T16987 CV7HN1 11795548 Ki = 7 nM T16987 C8DY3Z 11817193 IC50 = 7990 nM T16987 C73SVE 11817275 Ki = 6.7 nM T16987 C0CR2G 11848185 Ki = 12 nM T16987 C45NRP 11851425 Ki = 8.8 nM T16987 CZD0B3 11974341 Ki = 4.3 nM T16987 CC8AI5 11974342 Ki = 11.7 nM T16987 C27HSO 11974343 Ki = 8 nM T16987 CCM17V 11974451 Ki = 14.5 nM T16987 CX4IJ0 11974452 Ki = 19.7 nM T16987 C59UEI 11974453 Ki = 3.2 nM T16987 CYS7X0 11974454 Ki = 3.9 nM T16987 C09JGZ 11974455 Ki = 7.5 nM T16987 CS9VL2 11974456 Ki = 3.9 nM T16987 CP39YI 11974558 Ki = 6.1 nM T16987 CB97SM 11974559 Ki = 8.1 nM T16987 CE8WN6 11974560 Ki = 7.5 nM T16987 C06CBY 11974561 Ki = 7.4 nM T16987 CU6K0N 11974562 Ki = 1 nM T16987 CI7OE1 11974563 Ki = 14.7 nM T16987 C6Z5DX 11974630 Ki = 13.1 nM T16987 CW4X9G 11974631 Ki = 7.9 nM T16987 CEBO65 11974632 Ki = 7.7 nM T16987 C7TH2X 11974633 Ki = 7.6 nM T16987 CGQ6B7 11974724 Ki = 7.7 nM T16987 CHO9T1 11974725 Ki = 11.4 nM T16987 CB2DY9 11974726 Ki = 11.5 nM T16987 CC8TS1 11974727 Ki = 388 nM T16987 CDL18J 11974728 Ki = 7.1 nM T16987 CBC14R 11974729 Ki = 1.1 nM T16987 C7G3YS 11974830 Ki = 7.4 nM T16987 C1C4JW 11974831 Ki = 7.3 nM T16987 CXW89D 12004261 Ki = 30 nM T16987 C0L4OC 12049163 Ki = 37 nM T16987 CNHD71 12051191 Ki = 73000 nM T16987 CMPA32 12066940 Ki > 500000 nM T16987 CB15KR 12066941 Ki > 500000 nM T16987 C2XBZ3 12070806 Ki = 44 nM T16987 C32TWU 12094253 Ki = 67.6 nM T16987 C6P1VC 12188108 Ki = 9.4 nM T16987 C3C9ON 12226066 Ki = 800 nM T16987 CCY51E 12237458 Ki = 8.7 nM T16987 C60EFT 12354987 Ki = 940 nM T16987 CLB1E3 12499681 Ki = 673.5 nM T16987 CP87GR 12516475 Ki = 24.3 nM T16987 C5RS4H 12528487 Ki = 69.3 nM T16987 CM8TP6 12528490 Ki = 64.5 nM T16987 C35CMO 12589789 Ki = 64.7 nM T16987 CK90BP 12765315 Ki = 700 nM T16987 CO8WC5 12938307 Ki = 45.5 nM T16987 CF2BM7 13177311 Ki = 0.6 nM T16987 C8VM1A 13201770 Ki = 540 nM T16987 CV1UF4 13306723 Ki = 6.7 nM T16987 CX7M9C 13373975 Ki = 9.6 nM T16987 CHC41Q 13381193 Ki = 8.2 nM T16987 COLK69 13419352 Ki = 22.9 nM T16987 CFN29Y 13584466 Ki > 10000 nM T16987 CQTX49 13738810 IC50 = 350 nM T16987 CTYP72 13949092 Ki > 10000 nM T16987 CR6HB5 13949095 Ki > 10000 nM T16987 CFMK94 13949102 Ki > 10000 nM T16987 C7K4JV 14024589 Ki = 247.2 nM T16987 C4UG2O 14057643 Ki = 7390 nM T16987 CLS53V 14151811 IC50 = 464 nM T16987 CQ3D9C 14151815 IC50 = 461 nM T16987 C92OEB 14498136 Ki = 33 nM T16987 CHOG93 14611919 Ki = 110 nM T16987 CZ6SN8 14777102 Ki = 35.8 nM T16987 C76ASY 14787919 Ki > 200000 nM T16987 C35DGV 14873166 Ki = 7.1 nM T16987 C9CLH4 14873170 Ki > 10000 nM T16987 C9K0LX 14873174 Ki > 10000 nM T16987 CM34ER 14873177 Ki = 359.8 nM T16987 CH5YR2 15014351 Ki = 54500 nM T16987 C7XD2T 15118768 Ki = 770 nM T16987 CK8GE9 15230629 Ki = 764 nM T16987 C6F3GK 15267134 Ki = 6.3 nM T16987 CDE4F9 15290967 Ki = 292.4 nM T16987 CW72MS 15438999 Ki = 210 nM T16987 C7R5AH 15476112 Ki = 200 nM T16987 C3CTS0 15523879 Ki = 3.1 nM T16987 C2G4FH 15599374 Ki = 12.7 nM T16987 CLIO60 15645619 Ki = 5.5 nM T16987 C8PMQ9 15729847 Ki > 200000 nM T16987 CLT47Z 15783680 Ki = 56.4 nM T16987 C6F0XZ 15818962 Ki = 43.7 nM T16987 C8PER5 15938557 Ki > 500000 nM T16987 C3W2MB 15939939 Ki = 43.5 nM T16987 CB3S7I 16007202 Ki = 1.3 nM T16987 CM06OZ 16046226 Ki = 20 nM T16987 CVZG29 16072592 Ki = 14300 nM T16987 CB73ST 16072595 Ki = 9240 nM T16987 C6U0VS 16078349 Ki = 52 nM T16987 CUT32D 16078350 Ki > 1000 nM T16987 C4JIO0 16078351 Ki = 44 nM T16987 C23FGI 16078837 Ki = 170 nM T16987 CC74NH 16087011 Ki = 51.4 nM T16987 C1CD5B 16087012 Ki = 8.7 nM T16987 C8AP5W 16087015 Ki = 9.6 nM T16987 CLNI97 16087025 Ki = 10.1 nM T16987 CBWD20 16087028 Ki = 8.9 nM T16987 CN1XR0 16087029 Ki = 101 nM T16987 C3GMJ8 16087031 Ki = 13.1 nM T16987 CC0Z4V 16119626 Ki = 12700 nM T16987 CN03IT 16227153 Ki = 80.7 nM T16987 CGB45O 16235229 Ki = 181 nM T16987 CMB87O 16717602 Ki = 4.3 nM T16987 COQU32 16729004 Ki = 3 nM T16987 CTK68M 17249579 Ki = 2.5 nM T16987 C5DT7E 17250082 Ki = 7.9 nM T16987 C6THW2 17268490 Ki = 49.7 nM T16987 C5CE8Z 17371280 Ki = 0.57 nM T16987 CA4OE9 17371576 Ki = 0.65 nM T16987 C73YML 17385730 Ki = 9.9 nM T16987 C91LAN 17413757 Ki = 289 nM T16987 C5M9DR 17433209 Ki = 7.5 nM T16987 CYLM41 17492191 Ki = 9.3 nM T16987 CUP95O 17562622 Ki = 22.5 nM T16987 CLY1N4 17757567 Ki = 890 nM T16987 C6SFI8 18268734 Ki = 6.2 nM T16987 CR9VF3 18668331 Ki = 6.8 nM T16987 CQE5K4 18710120 Ki > 200000 nM T16987 C60NAV 18971452 Ki = 10.7 nM T16987 C2K5BX 19374444 Ki = 10.5 nM T16987 CIEH93 19382975 IC50 = 6917 nM T16987 C62PKT 19838794 Ki = 8.5 nM T16987 CU3QS7 19898674 Ki = 6.8 nM T16987 CB46JX 20109894 Ki = 7780 nM T16987 CGE35Q 20182298 Ki = 6.4 nM T16987 CDU40W 20184392 Ki = 3530 nM T16987 CXJ2H4 20195196 Ki = 4510 nM T16987 C15BEG 20694083 Ki = 49.5 nM T16987 CKR8T2 20970546 Ki = 8.6 nM T16987 CCJ8Q3 21051266 Ki = 52.8 nM T16987 CH15RE 21051367 Ki = 61.5 nM T16987 CJGU80 21240387 Ki = 28.3 nM T16987 C18KAH 21297028 Ki = 10.4 nM T16987 C9J1WT 21497848 Ki = 245 nM T16987 CC5W7X 21542156 Ki = 227 nM T16987 CD0K1C 21600238 Ki = 47 nM T16987 C61KUX 21726402 Ki = 0.79 nM T16987 CO2U7W 21855445 Ki = 5.4 nM T16987 CZ45AO 21878638 Ki = 40 nM T16987 C4XAO7 21879009 Ki = 18.1 nM T16987 CBS63Q 21879398 Ki = 53.6 nM T16987 C02IPY 21978067 Ki = 7.9 nM T16987 C6IZW0 22132896 Ki = 7.6 nM T16987 C9U4TE 22313850 Ki = 114 nM T16987 CPR25C 22706805 Ki = 630 nM T16987 C2D8ZL 23111570 Ki = 5.5 nM T16987 C2DOR4 23263451 Ki > 10000 nM T16987 C9KMP4 23275795 Ki = 2.5 nM T16987 CRZT32 23665339 Ki = 53.1 nM T16987 C7V6YP 23665706 Ki = 3.8 nM T16987 CXWP91 23666732 Ki = 0.99 nM T16987 C6W2BA 23668541 Ki = 709 nM T16987 CU08IW 23670409 Ki = 7.9 nM T16987 C1HCX5 23671974 Ki = 16.1 nM T16987 CDB01O 23674157 Ki = 7.5 nM T16987 CR7O3Q 23677931 Ki = 4.2 nM T16987 CKL59B 23679442 Ki = 6 nM T16987 CC93FA 23686905 Ki = 11.5 nM T16987 CZD6O0 23688497 Ki = 75.6 nM T16987 CE91KL 23691977 Ki = 561 nM T16987 CK2Q0I 23697126 Ki = 15.3 nM T16987 CPX0I4 24204718 Ki = 29 nM T16987 CF83JT 24204719 Ki = 36 nM T16987 CSWR58 24204720 Ki = 24 nM T16987 CIQ9L6 24204924 Ki = 28 nM T16987 CL2V5T 24204925 Ki = 29 nM T16987 C14RLU 24204932 Ki = 27 nM T16987 CN5ST6 24206002 Ki = 24 nM T16987 CPD4Z6 24206003 Ki = 14 nM T16987 C1Y2JB 24286289 Ki = 7 nM T16987 CKE1A3 24416843 Ki = 0.93 nM T16987 CGHW54 24640576 Ki = 3.5 nM T16987 C01LHS 24640776 Ki = 2.7 nM T16987 CT8O2Z 24643222 Ki = 7.3 nM T16987 CB6WE3 24650532 Ki = 91.4 nM T16987 C1I9HZ 24692821 Ki = 2.7 nM T16987 CQG9O0 24816432 Ki = 19 nM T16987 CK0D4U 24823300 Ki = 40.1 nM T16987 C5W7AC 24823303 Ki = 67.1 nM T16987 CZMT56 24823304 Ki = 9.7 nM T16987 CUT3V8 24823479 Ki = 36.3 nM T16987 CNR3U7 24866945 IC50 > 10000 nM T16987 CQRZ10 24877657 Ki = 4.2 nM T16987 C62DIS 25048179 Ki = 90.3 nM T16987 COI25U 25131351 Ki = 30 nM T16987 CNMY17 25131685 Ki = 147 nM T16987 CISH83 25186263 Ki = 5.7 nM T16987 CU14KG 25258358 Ki = 65000 nM T16987 CQ1WE2 25258360 Ki = 70800 nM T16987 CL5EZ6 25258361 Ki = 65400 nM T16987 COU19V 25258363 Ki = 61200 nM T16987 C5T1NZ 25294048 Ki = 67.4 nM T16987 CPN2T5 25392418 Ki = 86.6 nM T16987 C1AOB3 25981084 Ki = 4.6 nM T16987 CP02LF 26365005 Ki = 3.9 nM T16987 C0RF4D 26470767 Ki = 184 nM T16987 CMUT78 26500397 Ki = 3.5 nM T16987 C5EC2T 26535209 Ki = 3.8 nM T16987 CLNR46 26598995 Ki = 325.7 nM T16987 CA9UZ7 26773685 Ki = 3.1 nM T16987 C8KQ5N 27868059 Ki = 7.1 nM T16987 CQSA29 27868075 Ki = 6.2 nM T16987 C7QB8M 27868953 Ki = 179 nM T16987 CWU2R0 27869227 Ki = 113 nM T16987 C46OQT 27869236 Ki = 149 nM T16987 C85HLF 27869237 Ki = 48.6 nM T16987 C5OWP7 27869350 Ki = 64.5 nM T16987 CF02EA 27869546 Ki = 165 nM T16987 C1G3XO 27869982 Ki = 7.9 nM T16987 C8ML3W 27870055 Ki = 4.3 nM T16987 CMK25I 27870443 Ki = 7 nM T16987 CQK4O6 27870796 Ki = 4.6 nM T16987 C2Z4FP 27870803 Ki = 39 nM T16987 C3RG8K 28846439 Ki = 11.5 nM T16987 C4EB0J 29034199 Ki = 21 nM T16987 CF8SA7 29559803 Ki = 138 nM T16987 CF3HA1 35871284 Ki = 16.4 nM T16987 CI0K1J 36865965 Ki = 7.9 nM T16987 C5IUO9 38154971 Ki = 113 nM T16987 CZE95V 38155699 Ki = 96.4 nM T16987 CSB4C7 38159448 Ki = 66.9 nM T16987 C4F7YT 40086402 Ki = 6 nM T16987 C06EUO 40662472 Ki = 10.5 nM T16987 C1U4TL 41180562 Ki = 63 nM T16987 CH2P6W 41430216 Ki = 28.5 nM T16987 C5YBO2 41484755 Ki = 55.4 nM T16987 CUK13R 41874556 Ki = 8 nM T16987 C0J8DM 42597612 Ki = 4710 nM T16987 C8A5CF 42597613 Ki = 4800 nM T16987 C58ZUN 42597614 Ki = 4770 nM T16987 COG2A0 42597615 Ki = 4600 nM T16987 C1J9CQ 42597616 Ki = 4550 nM T16987 COG2I5 42598921 Ki = 4610 nM T16987 CDXS12 42598922 Ki = 4840 nM T16987 C6WU8M 42609905 Ki = 0.36 nM T16987 CYJ0H4 43089860 Ki = 4.5 nM T16987 CXJY80 43235186 Ki = 7.8 nM T16987 C7EO2A 43329592 Ki = 6.4 nM T16987 CA0DX4 43342474 Ki = 8 nM T16987 C2HY4R 43342475 Ki = 1.2 nM T16987 CBK0M6 43342481 Ki = 0.72 nM T16987 C41VHR 43468983 Ki = 0.71 nM T16987 C82MRL 44144383 Ki = 17.8 nM T16987 CVJ5A1 44246262 Ki = 6.1 nM T16987 CZKG76 44246264 Ki = 6.3 nM T16987 C3E0CZ 44246268 Ki = 7.9 nM T16987 C0QZI4 44246269 Ki = 7.2 nM T16987 CZL01D 44246271 Ki = 7.4 nM T16987 C91HDR 44315566 Ki = 736.3 nM T16987 C5O9LH 44389667 Ki = 3 nM T16987 CL5GF2 44389703 Ki = 1.9 nM T16987 C9DRN1 44389734 Ki = 4.9 nM T16987 CE9BS6 44389758 Ki = 1.7 nM T16987 C68TCP 44389772 Ki = 2.3 nM T16987 C9OM5F 44389791 Ki = 2.1 nM T16987 C7VMQ6 44389836 Ki = 33 nM T16987 CF19RI 44389844 Ki = 50 nM T16987 CG2U5A 44389881 Ki = 10 nM T16987 CR16DV 44389954 Ki = 24 nM T16987 C8KE4X 44389960 Ki = 13 nM T16987 CEV89Z 44389961 Ki = 1.8 nM T16987 C5ZCF3 44389968 Ki = 12 nM T16987 C06AUB 44389978 Ki = 2 nM T16987 C09EFT 44389990 Ki = 1.5 nM T16987 CFBU06 44389993 Ki = 12 nM T16987 C3IBQ1 44389995 Ki = 4.8 nM T16987 CP8JK3 44390019 Ki = 3 nM T16987 CWCQ49 44390027 Ki = 144 nM T16987 CVW6E1 44390031 Ki = 3.3 nM T16987 C5TO9D 44390032 Ki = 64 nM T16987 CD9H6W 44392389 Ki = 3.4 nM T16987 C9J2ME 44395133 Ki = 43.8 nM T16987 CI3O9B 44395149 Ki = 22.7 nM T16987 CPB8W7 44395163 Ki = 56.2 nM T16987 CMSJ40 44395790 Ki = 3.1 nM T16987 C5GJ3N 44399351 Ki = 2.9 nM T16987 CZ4DF9 44399462 Ki = 2.6 nM T16987 CU7BK9 44399535 Ki = 3.5 nM T16987 CD5MJ6 44399571 Ki = 10.2 nM T16987 C2T7MB 44399654 Ki = 8.9 nM T16987 CT6UF5 44402709 Ki = 38 nM T16987 C5FC0Y 44402716 Ki > 1000 nM T16987 C8N0GW 44402748 Ki = 50 nM T16987 C9AJ7Z 44402772 Ki = 33 nM T16987 CR72VG 44402825 Ki = 27 nM T16987 C6OS3R 44403265 Ki = 2.4 nM T16987 CSN79Y 44403312 Ki = 76 nM T16987 CVJ5T9 44416166 Ki = 35.6 nM T16987 CZT1U9 44416167 Ki > 10000 nM T16987 CQ36IP 44416168 Ki = 53 nM T16987 CS49FE 44416185 Ki = 2404 nM T16987 CEH5P1 44416186 Ki = 3045 nM T16987 C8C4IJ 44416203 Ki > 10000 nM T16987 CE6N7Q 44416215 Ki > 10000 nM T16987 CY9VT1 44416239 Ki = 117 nM T16987 CI01QM 44416240 Ki = 108 nM T16987 CX8ZQ9 44416241 Ki = 1000 nM T16987 CRX27F 44416256 Ki = 1970 nM T16987 C68YLB 44416306 Ki = 1103 nM T16987 C5ROE2 44416307 Ki = 1390 nM T16987 C47OTU 44416317 Ki = 2417 nM T16987 CE4M9P 44416378 Ki = 190 nM T16987 CE03DL 44416379 Ki > 10000 nM T16987 CA90GQ 44424362 Ki = 770 nM T16987 C5HB4P 44424363 Ki > 200000 nM T16987 CK8S7Y 44424364 Ki > 200000 nM T16987 C28QYE 44424366 Ki = 910 nM T16987 CP3OY8 44428369 Ki = 33.9 nM T16987 CQUC34 44520900 Ki = 12 nM T16987 CHCT21 44542292 Ki = 8.2 nM T16987 CG61YX 44542293 Ki = 9.9 nM T16987 CL8AQ5 44542294 Ki = 7.9 nM T16987 CF2RX4 44542600 Ki = 5.9 nM T16987 C5MZ3O 44542742 Ki = 7.6 nM T16987 CI9VZ6 44542743 Ki = 7.5 nM T16987 CKT85S 44577800 Ki = 6 nM T16987 C3DU8S 44577801 Ki = 3.6 nM T16987 CCW3S1 44578981 Ki = 128 nM T16987 CU7Y8T 44578982 Ki = 78 nM T16987 C86YLD 44579460 Ki = 55 nM T16987 CD4WO8 44579535 Ki = 6 nM T16987 CXD9V3 44590306 Ki = 56300 nM T16987 CM2L4W 44591861 Ki = 9.4 nM T16987 CQ40FB 44592373 Ki = 9.5 nM T16987 C15THP 44592446 Ki = 8.4 nM T16987 CDB3X7 44592447 Ki = 9.1 nM T16987 C2J3ER 44592448 Ki = 9.2 nM T16987 CUXJ39 44592449 Ki = 9.5 nM T16987 CTI2C1 44592450 Ki = 10.9 nM T16987 COS6N0 44592512 Ki = 9.5 nM T16987 CASL51 44592513 Ki = 10.2 nM T16987 CXL68J 44592514 Ki = 10.3 nM T16987 COL03N 44592515 Ki = 10.3 nM T16987 CHMW14 44592516 Ki = 11.9 nM T16987 COX6D8 45028566 Ki = 7.8 nM T16987 CF2WL9 45028890 Ki = 113 nM T16987 C4MO3S 45028891 Ki = 75 nM T16987 C80CDA 45028892 Ki = 6.1 nM T16987 C6YHW4 45028893 Ki = 8.7 nM T16987 C16ILW 45028894 Ki = 34.6 nM T16987 COE8U0 45267045 Ki = 453.6 nM T16987 CA07CZ 45268031 Ki = 73 nM T16987 C23MVW 45269009 IC50 = 48600 nM T16987 C0RG8K 45269749 Ki = 8700 nM T16987 C6E7XJ 45484068 Ki = 4660 nM T16987 CGI25L 45484069 Ki = 4710 nM T16987 CVG6K1 45484072 Ki = 4690 nM T16987 CV5RQ3 45484187 Ki = 9500 nM T16987 CTG20B 45485271 Ki = 42000 nM T16987 CK4U0V 45485283 Ki = 15600 nM T16987 C5GZ1B 46197458 Ki = 11.5 nM T16987 C3Z7OL 46197569 Ki = 15.5 nM T16987 CUQF42 46197571 Ki = 9.8 nM T16987 C4C7XG 46197572 Ki = 8.5 nM T16987 CLBG91 46197677 Ki = 9.3 nM T16987 C9GC5Q 46197678 Ki = 9.9 nM T16987 C16XCV 46197680 Ki = 10.4 nM T16987 C3JW1R 46197790 Ki = 9.1 nM T16987 CD49XQ 46197791 Ki = 8.3 nM T16987 C4H9TD 46197792 Ki = 8.7 nM T16987 C0W1GZ 46197794 Ki = 8.9 nM T16987 CUO20Q 46197893 Ki = 8.2 nM T16987 CN7KI3 46197894 Ki = 13.6 nM T16987 CD74LO 46197895 Ki = 16.7 nM T16987 CZ93SW 46197897 Ki = 8.7 nM T16987 CNQZ73 46197997 Ki = 8.8 nM T16987 CCAX25 46197998 Ki = 9.5 nM T16987 CQ3R2U 46197999 Ki = 9.4 nM T16987 CGM42H 46198111 Ki = 9.5 nM T16987 C0DKY8 46198112 Ki = 8.8 nM T16987 CBWN61 46198113 Ki = 7.6 nM T16987 C0AF1L 46198114 Ki = 7.8 nM T16987 C1KWB5 46198220 Ki = 9.1 nM T16987 CEV26X 46198221 Ki = 7.3 nM T16987 C25FBC 46567082 Ki = 31.6 nM T16987 CA4FJ2 46703925 Ki = 4.2 nM T16987 C2WB4C 46703927 Ki = 21.6 nM T16987 CO2IU4 46704079 Ki = 15.1 nM T16987 CB85EQ 46704080 Ki = 3.4 nM T16987 CAE9Z3 46704081 Ki = 8.1 nM T16987 CD5V6T 46704082 Ki = 4.6 nM T16987 C8MR0H 46847340 IC50 = 6200 nM T16987 CRS8J6 46860267 Ki = 6 nM T16987 C2RA7G 46861342 Ki = 24.5 nM T16987 C2S4YC 46866644 IC50 = 6900 nM T16987 C7QR8Y 46866645 IC50 = 6400 nM T16987 CUH07J 46866646 IC50 = 5600 nM T16987 C8GK4C 46866647 IC50 = 5700 nM T16987 CT65RE 46868356 Ki = 228.4 nM T16987 C7UKN2 46884029 Ki = 15.6 nM T16987 C1DCM9 46884093 Ki = 9.8 nM T16987 C4ALG9 46884132 Ki = 8.9 nM T16987 CTRY21 46884169 Ki = 9.5 nM T16987 CBM20W 46884215 Ki = 9.7 nM T16987 CR61DW 46884254 Ki = 9.5 nM T16987 C93AIR 46899573 Ki = 112000 nM T16987 C4GZ6A 46907387 Ki = 5.1 nM T16987 CJ0R2O 46911381 Ki = 4.7 nM T16987 C9T3WF 46933594 Ki = 146 nM T16987 C1WE2D 46933744 Ki = 35.6 nM T16987 CUHI56 46933745 Ki = 32.5 nM T16987 C27DFQ 46933746 Ki = 25.4 nM T16987 CSQG87 46933747 Ki = 31.8 nM T16987 C08BKN 46933748 Ki = 12.2 nM T16987 C54PRX 46933749 Ki = 127 nM T16987 CP62AV 46933896 Ki = 381 nM T16987 C03FQY 46943413 Ki = 29.7 nM T16987 CCOB94 49929067 Ki = 404 nM T16987 C5Z2QA 50741845 Ki = 6.6 nM T16987 CVC35K 50899076 IC50 = 7640 nM T16987 CR3I2H 50899077 IC50 = 5430 nM T16987 CEHP41 50909907 Ki = 5.7 nM T16987 CB4O0Y 50909908 Ki = 4.2 nM T16987 C1QBZ3 50942416 Ki = 2.5 nM T16987 C62ZDQ 51035422 Ki = 1.6 nM T16987 CW0CJ2 51035423 Ki = 6.7 nM T16987 C5CR2F 51039206 Ki = 8.4 nM T16987 C3SH7R 51039207 Ki = 7.6 nM T16987 CS5ZR3 51039209 Ki = 93 nM T16987 C8TR3Z 51047320 Ki = 213 nM T16987 CHK5G9 51059586 Ki = 2010 nM T16987 C8XGV5 51349458 Ki = 85 nM T16987 C4S5NC 51349459 Ki = 96 nM T16987 CZH4T2 51349599 Ki = 87 nM T16987 CK3U6Q 51349600 Ki = 9.5 nM T16987 CDF2V8 51349601 Ki = 145 nM T16987 CG26DK 51349604 Ki = 138 nM T16987 CUP39M 51355749 Ki = 52.8 nM T16987 CJ1M5T 51355750 Ki = 6.5 nM T16987 CBL9U1 51356010 Ki = 65.1 nM T16987 CLG43P 51669707 IC50 = 8260 nM T16987 CPGW70 53245686 Ki = 31 nM T16987 CCW69Q 53308637 Ki = 78 nM T16987 CKRO12 53321135 Ki = 9.5 nM T16987 CTF92V 53322463 Ki = 7.3 nM T16987 C8Z2IL 53324362 Ki = 7.6 nM T16987 CK4ZG3 53342705 Ki = 2 nM T16987 CHF62Q 53361485 IC50 = 386 nM T16987 CJ3F4R 53361486 IC50 = 476 nM T16987 C08REF 53364160 Ki = 4.8 nM T16987 C32UEX 53364161 Ki = 7.8 nM T16987 CHWX25 53364162 Ki = 5.6 nM T16987 C58YMC 53371608 Ki = 19 nM T16987 C0NUM6 53386724 Ki = 9.1 nM T16987 C54FGU 53386866 Ki = 10.5 nM T16987 CRI54V 53386867 Ki = 8.6 nM T16987 CUX7S4 53386868 Ki = 25.3 nM T16987 CSA60L 53389267 Ki = 58.9 nM T16987 C8VXD9 53389268 Ki = 0.8 nM T16987 CV40HR 53426278 Ki = 52.3 nM T16987 C6T5RC 53483944 Ki = 1.2 nM T16987 CM5KX6 53483945 Ki = 9.2 nM T16987 C3M4EL 53483958 Ki = 12 nM T16987 CY2MI0 54077127 Ki = 798 nM T16987 CB6W4D 54577841 Ki = 8 nM T16987 CHCT45 54580732 Ki = 29 nM T16987 CYB47X 54581736 Ki = 43 nM T16987 CW2KI4 54582723 Ki = 31 nM T16987 CWK6B0 54582724 Ki = 116 nM T16987 CBS8R1 54584666 Ki = 42 nM T16987 CJ3UE2 54584667 Ki = 87 nM T16987 CO0BD9 54585508 Ki = 83 nM T16987 C0A5OZ 54612935 Ki = 28.5 nM T16987 C6X7QG 54613732 Ki = 9.9 nM T16987 CKB0G9 54669765 Ki = 10 nM T16987 CS8IV7 54669781 Ki = 10.7 nM T16987 C0PJ1K 54677403 Ki = 453.5 nM T16987 CAS91K 54682930 Ki = 6300 nM T16987 CQ3XK0 54758050 Ki = 8.9 nM T16987 C5ON9E 54758136 Ki = 8.6 nM T16987 C0K2LN 54758137 Ki = 9.1 nM T16987 C5Q9XC 54758138 Ki = 59.2 nM T16987 CLT0W2 54758232 Ki = 53.1 nM T16987 C5V4GI 54758233 Ki = 7.8 nM T16987 C98JVL 54758234 Ki = 5.3 nM T16987 CXBF42 54758235 Ki = 9.4 nM T16987 C4EL5V 54758236 Ki = 11.7 nM T16987 CU19DH 54758322 Ki = 56 nM T16987 CE53AN 54758323 Ki = 7.9 nM T16987 CK3Q0O 54758324 Ki = 9 nM T16987 CE2O3A 54768697 Ki = 7.5 nM T16987 C5SB4M 54768698 Ki = 9.1 nM T16987 CBNP25 54768699 Ki = 6 nM T16987 C9Z4RJ 54772055 Ki = 16.4 nM T16987 CB3EC8 54772057 Ki = 8.2 nM T16987 CE6LD4 54772059 Ki = 9 nM T16987 CD5P1I 54772061 Ki = 9.9 nM T16987 C0ZJ2L 55629711 Ki > 50000 nM T16987 CK89GH 56659335 Ki = 8.7 nM T16987 C05JRQ 56659336 Ki = 9.2 nM T16987 CEC29W 56659337 Ki = 8.6 nM T16987 C2TW1F 56659553 Ki = 6.4 nM T16987 CO9SW8 56659554 Ki = 78 nM T16987 CVRM21 56659555 Ki = 7 nM T16987 CJ43WP 56659826 Ki = 5440 nM T16987 CZ4HI1 56662794 Ki = 8.5 nM T16987 CD8SR3 56662795 Ki = 43.9 nM T16987 CF0J6I 56663002 Ki = 7 nM T16987 CH0MV2 56663442 Ki = 9.4 nM T16987 CM07OK 56663443 Ki = 57 nM T16987 CVM8W4 56666268 Ki = 6 nM T16987 C89SEG 56666269 Ki = 20.7 nM T16987 C36TYE 56666270 Ki = 7.1 nM T16987 CD5OZ4 56666482 Ki = 6.3 nM T16987 CI93KS 56666719 Ki = 8230 nM T16987 CR9F8U 56670316 Ki = 59 nM T16987 CF1J7H 56670317 Ki = 86 nM T16987 CWNF20 56673403 Ki = 79 nM T16987 CT29KP 56673404 Ki = 81 nM T16987 C7DU3M 56673405 Ki = 7.8 nM T16987 CHV04E 56673655 Ki = 5.8 nM T16987 C4YI1B 56673656 Ki = 1970 nM T16987 CKL09N 56673817 Ki = 410 nM T16987 CI2R9B 56676517 Ki = 0.85 nM T16987 C9X7VM 56676518 Ki = 5.8 nM T16987 CF86WB 56676713 Ki = 6.9 nM T16987 CDH07V 56677155 Ki = 104 nM T16987 CR7D6S 56677156 Ki = 10 nM T16987 C2U1VF 56679839 Ki = 9.3 nM T16987 CS81JH 56680034 Ki = 7.1 nM T16987 C02WBE 56680461 Ki = 76 nM T16987 CEZ3F5 56683163 Ki = 248 nM T16987 C4LB1M 56683164 Ki = 80 nM T16987 CZS9V5 56683165 Ki = 82 nM T16987 C8V1PA 56683626 Ki = 6.5 nM T16987 CXL7Q1 56683627 Ki = 9900 nM T16987 CIJ9V0 56684131 Ki = 5870 nM T16987 CTWZ62 56836370 Ki = 7.4 nM T16987 C49PBJ 56836371 Ki = 6.2 nM T16987 CK7Y8J 56836443 Ki = 78.5 nM T16987 CY7Z1A 56836444 Ki = 83.6 nM T16987 CV0ST7 56836445 Ki = 10.1 nM T16987 C0O3UI 56836446 Ki = 8.5 nM T16987 C0PKB5 56836447 Ki = 6.4 nM T16987 CZ9F7P 56836511 Ki = 8.3 nM T16987 COY29V 56836512 Ki = 6.8 nM T16987 C7PWG1 56836513 Ki = 6.1 nM T16987 C4CF8M 56836514 Ki = 8.2 nM T16987 C4IRK8 56836515 Ki = 7.6 nM T16987 CH52DA 56921864 Ki = 6490 nM T16987 C0Z8WY 56925533 Ki = 101 nM T16987 CC3Q9S 56928516 Ki = 67.1 nM T16987 CO18AP 57011620 Ki = 6.7 nM T16987 C4VGE9 57047254 Ki = 4.1 nM T16987 CNG76Q 57326130 Ki = 9.2 nM T16987 C81YCD 57326131 Ki = 17.5 nM T16987 C4TV1U 57326132 Ki = 31.7 nM T16987 CHL0B3 57326133 Ki = 4.2 nM T16987 C5Z4SW 57326134 Ki = 9.3 nM T16987 CFU62Y 57326227 Ki = 20.5 nM T16987 C97HYX 57326228 Ki = 6.5 nM T16987 CS4I5T 57326229 Ki = 4 nM T16987 CP7YR5 57345662 Ki = 64 nM T16987 C0S2YZ 57383964 Ki = 12.5 nM T16987 C97GHV 57383965 Ki = 9.8 nM T16987 CXW5D3 57384052 Ki = 280 nM T16987 C4XF9A 57384114 Ki = 10.1 nM T16987 CS76WU 57384115 Ki = 8.2 nM T16987 C0UBL5 57384116 Ki = 8.6 nM T16987 C16AGY 57384117 Ki = 8.5 nM T16987 CVWK43 57386884 Ki = 830 nM T16987 CR3C7D 57386885 Ki = 310 nM T16987 C9CX4B 57386886 Ki = 350 nM T16987 CZOD69 57386887 Ki = 340 nM T16987 CZN72E 57386888 Ki = 1270 nM T16987 C9JU0H 57386889 Ki = 1250 nM T16987 CQ0I4V 57386890 Ki = 900 nM T16987 C8Z0DJ 57387135 Ki = 590 nM T16987 C1HZS5 57387136 Ki = 640 nM T16987 C7EN6Z 57387137 Ki = 580 nM T16987 C87ASQ 57387395 Ki = 38900 nM T16987 CQW5T3 57387397 Ki = 370 nM T16987 CT3B0Z 57387636 Ki = 2830 nM T16987 C09GQI 57392249 Ki = 7.2 nM T16987 CY81SU 57392250 Ki = 7.8 nM T16987 CMEV16 57392251 Ki = 8.4 nM T16987 C94YIX 57392252 Ki = 8.2 nM T16987 CM7S3H 57394009 Ki = 7.3 nM T16987 CHAF57 57394010 Ki = 7.6 nM T16987 CV7K9Y 57394771 Ki = 20.1 nM T16987 CM4SL9 57394772 Ki = 81 nM T16987 C1M0LS 57394809 Ki = 760 nM T16987 CJ5XK2 57395770 Ki = 8.9 nM T16987 CV6QX4 57395771 Ki = 8.8 nM T16987 CHG91B 57396529 Ki = 10.2 nM T16987 C9H4VS 57396530 Ki = 8.7 nM T16987 C6XD2O 57397549 Ki = 8.4 nM T16987 C64VIW 57397550 Ki = 8.1 nM T16987 CRIU35 57398318 Ki = 8.2 nM T16987 CN6TU2 57398319 Ki = 13.5 nM T16987 C97OJM 57399231 Ki = 7.5 nM T16987 C7XAZ3 57399232 Ki = 48.1 nM T16987 CK24NA 57399233 Ki = 9.7 nM T16987 CG3X4V 57401764 Ki = 7.9 nM T16987 C4V5KY 57402747 Ki = 45.6 nM T16987 CRU53E 57402748 Ki = 100 nM T16987 C52TUM 57402749 Ki = 8.2 nM T16987 CQ9ZG2 57402750 Ki = 7.4 nM T16987 C80WTZ 57403496 Ki = 111 nM T16987 CDIM87 57403497 Ki = 300 nM T16987 C76ZDS 57404539 Ki = 7.7 nM T16987 CKID78 57411990 Ki = 2.7 nM T16987 C4ZYF3 57411991 Ki = 3.1 nM T16987 CDG6R4 57411992 Ki = 5 nM T16987 CKPS17 57411993 Ki = 4.7 nM T16987 CV13LT 57411994 Ki = 58 nM T16987 C5JDQ1 57413825 Ki = 64 nM T16987 C5M4CN 57413826 Ki = 8 nM T16987 C3D7KS 57413827 Ki = 8.1 nM T16987 CJO26X 57413828 Ki = 6.7 nM T16987 CA4CD7 57413968 Ki = 8.1 nM T16987 CQ1ZK6 57519697 Ki = 57 nM T16987 CG3W0D 58404071 Ki = 59 nM T16987 CT3B7P 58477593 Ki = 5.53 nM T16987 C01TQW 59079460 Ki = 7.4 nM T16987 CF1NG0 60155028 Ki = 3.679 nM T16987 C0PRW7 60155029 Ki = 3.934 nM T16987 CNX97Q 60155030 Ki = 3 nM T16987 CR0Z7W 60155031 Ki = 3.73 nM T16987 CI2WL7 60155120 Ki = 1 nM T16987 CM57BF 60155121 Ki = 3.788 nM T16987 C5VF9X 60155122 Ki = 4 nM T16987 C2U8VH 60155123 Ki = 2 nM T16987 CNR53M 60155124 Ki = 29 nM T16987 CYQM98 60201413 Ki = 54 nM T16987 CGWU14 60201414 Ki = 580 nM T16987 C6TP2W 60201415 Ki = 62 nM T16987 C1JVP9 60201416 Ki = 53 nM T16987 CQZN79 60201417 Ki = 48 nM T16987 CVU0B4 60201577 Ki = 79 nM T16987 CS3N6M 60201578 Ki = 0.5 nM T16987 CB45GM 60201579 Ki = 3.9 nM T16987 C1CVG9 61580845 Ki = 90.5 nM T16987 C9UD2V 62141270 Ki = 965.7 nM T16987 CZ4BQ6 66571808 Ki = 6.7 nM T16987 CGB46T 66571809 Ki = 8.2 nM T16987 CT0S3A 66572208 Ki = 8.9 nM T16987 CGF3W6 66586679 Ki = 890 nM T16987 CN84CU 66586879 Ki = 820 nM T16987 C54HCL 68341722 Ki = 7.9 nM T16987 C4MB5P 68602550 Ki = 151 nM T16987 CV6PY2 68833705 Ki = 47 nM T16987 C23JZS 70037678 Ki = 67 nM T16987 C6RVC3 70202738 Ki = 81.2 nM T16987 CDO92J 70681983 Ki = 3.633 nM T16987 CHC54M 70681984 Ki = 3.934 nM T16987 C1FY3K 70681985 Ki = 3.679 nM T16987 CSW7I0 70681986 Ki = 3.633 nM T16987 CP65RU 70681987 Ki = 2.863 nM T16987 CFT68C 70681988 Ki = 4 nM T16987 CR0D9S 70684100 Ki = 3 nM T16987 CRZ8S1 70684101 Ki = 3.934 nM T16987 COS95H 70684102 Ki = 4 nM T16987 CT5PH1 70684103 Ki = 3.378 nM T16987 C9P4BK 70685635 Ki = 169 nM T16987 C5XTY9 70686245 Ki = 3.934 nM T16987 C4SCY0 70688360 Ki = 2.971 nM T16987 CPD1N7 70688361 Ki = 2.97 nM T16987 C4L2OE 70688362 Ki = 3.218 nM T16987 CZO9C5 70688363 Ki = 3.171 nM T16987 CAD39I 70688364 Ki = 3.236 nM T16987 C7N4RT 70690386 Ki = 3.73 nM T16987 CQD8R9 70690387 Ki = 3.934 nM T16987 C1T4JL 70690936 Ki = 770 nM T16987 CUY3O8 70690937 Ki = 12800 nM T16987 CXF59L 70692549 Ki = 3.633 nM T16987 CV76WB 70692550 Ki = 3.855 nM T16987 C89LCZ 70692551 Ki = 3.378 nM T16987 C1K8VS 70692552 Ki = 3.855 nM T16987 CO5JP7 70692553 Ki = 3.855 nM T16987 CK5Y7G 70692554 Ki = 3.52 nM T16987 CGD06J 70692555 Ki = 3.592 nM T16987 C5QOK4 70692556 Ki = 3.487 nM T16987 C4BDK3 70694601 Ki = 2 nM T16987 CW8YA7 70694602 Ki = 2.741 nM T16987 CCYE61 70694603 Ki = 3.855 nM T16987 CEF1J8 70694604 Ki = 3.065 nM T16987 C4C0HK 70694605 Ki = 3 nM T16987 CBDQ72 70694606 Ki = 3 nM T16987 C95YWO 70695124 Ki = 3240 nM T16987 CSH7P1 70696148 Ki = 7.5 nM T16987 CWSA94 70696638 Ki = 3.73 nM T16987 CREC06 70696639 Ki = 3.855 nM T16987 CJ4M9S 70696640 Ki = 3.554 nM T16987 CHFY23 70696641 Ki = 3.934 nM T16987 C3Z7ER 70696642 Ki = 2.795 nM T16987 C6E4UW 70696643 Ki = 4 nM T16987 C0SP9E 70696644 Ki = 4 nM T16987 CAFH02 70696645 Ki = 4 nM T16987 CWQM13 70696646 Ki = 2 nM T16987 C04HIK 70698419 Ki = 4510 nM T16987 C8FB0P 71273627 Ki = 2.901 nM T16987 CJH6Y7 71273628 Ki = 3.554 nM T16987 CXG0H9 71273629 Ki = 3.218 nM T16987 CUT6R1 71273630 Ki = 3.934 nM T16987 CH49BT 71273631 Ki = 3.186 nM T16987 CK2U8R 71273632 Ki = 3.73 nM T16987 C2F9PC 71273633 Ki = 3.077 nM T16987 CV8FW3 71273635 Ki = 2.253 nM T16987 CQJ61A 71273738 Ki = 2.642 nM T16987 CSMV41 71273739 Ki = 3.429 nM T16987 CYW59B 71273740 Ki = 3.236 nM T16987 CU0KV6 71273743 Ki = 3.73 nM T16987 CC21VR 71273744 Ki = 3.73 nM T16987 C80KUG 71273750 Ki = 3.679 nM T16987 CJHN78 71415156 Ki = 1427 nM T16987 C16PMU 71449958 IC50 = 2720 nM T16987 CXJ16H 71450117 Ki = 5540 nM T16987 CR79UB 71450332 Ki = 62.9 nM T16987 CT8E7N 71451561 Ki = 43 nM T16987 CHI2Z6 71452138 Ki = 79.8 nM T16987 CNI0R5 71452603 Ki = 45.2 nM T16987 C4E6PS 71453593 IC50 = 8600 nM T16987 CP27AT 71453970 Ki = 40.5 nM T16987 CW49YT 71453971 Ki = 43.3 nM T16987 C52WNJ 71454366 Ki = 81.8 nM T16987 CB8JA3 71455488 Ki = 6755 nM T16987 C02UHX 71455489 Ki = 4550 nM T16987 CZ0S7D 71455712 Ki = 73.7 nM T16987 CUX07I 71455715 Ki = 47.2 nM T16987 C9COK3 71456113 Ki = 58 nM T16987 CICJ97 71457274 Ki = 5620 nM T16987 CL2BN6 71457492 Ki = 75.4 nM T16987 C4L0BG 71457918 Ki = 70.6 nM T16987 CWHN25 71459359 Ki = 81.6 nM T16987 CE31LC 71459360 Ki = 70.5 nM T16987 C70MBK 71459826 Ki = 66.3 nM T16987 C95MKT 71459827 Ki = 73.8 nM T16987 C5WYI8 71459828 Ki = 72.4 nM T16987 CD93TU 71461134 Ki = 73.1 nM T16987 C3WKX5 71461135 Ki = 68.4 nM T16987 C3YSR8 71461136 Ki = 32.4 nM T16987 CS1WI7 71461542 Ki = 23.5 nM T16987 C7VQ1R 71461543 Ki = 36.9 nM T16987 C4X1BZ 71462495 IC50 = 6020 nM T16987 CUM2H8 71462868 Ki = 82.3 nM T16987 CU4N0L 71462869 Ki = 26.5 nM T16987 C9KZA2 71462872 Ki = 61.3 nM T16987 CI6V9W 71489159 Ki = 570 nM T16987 CMHG14 71521493 Ki = 6200 nM T16987 CHN53G 71521494 Ki = 3900 nM T16987 CZJ5M6 71521495 Ki = 4200 nM T16987 CFBE53 71521496 Ki = 7400 nM T16987 CME27W 71521497 Ki = 8400 nM T16987 C24XWU 71521575 Ki = 6700 nM T16987 CJF68W 71521576 Ki = 6800 nM T16987 CHL8P3 71522144 Ki = 23 nM T16987 CEYG83 71522162 Ki = 3160 nM T16987 CZ78YT 71522163 Ki = 2930 nM T16987 C8NAF3 71545047 Ki = 32 nM T16987 C4H6PD 71545048 Ki = 12 nM T16987 CQ20AS 71545049 Ki = 13 nM T16987 CG2CL6 71545050 Ki = 9 nM T16987 C1MET8 71545051 Ki = 16 nM T16987 CILC35 71545052 Ki = 7 nM T16987 CGQ97W 71545216 Ki = 14 nM T16987 C71UMX 71545217 Ki = 39 nM T16987 C3KJ6D 71545218 Ki = 13 nM T16987 C0JNF3 71545219 Ki = 21 nM T16987 CC5EB7 71570660 Ki = 2.16 nM T16987 CA82YW 71570661 Ki = 0.68 nM T16987 CNL58G 71570662 Ki = 3.48 nM T16987 CDGY15 71578422 Ki = 50.5 nM T16987 CA5M6S 71578423 Ki = 71.5 nM T16987 CGOR42 71578424 Ki = 19 nM T16987 C45YXJ 71578425 Ki = 34.9 nM T16987 C1CKL6 71578426 Ki = 31.4 nM T16987 CR38IX 71578427 Ki = 32 nM T16987 CQ8Z5T 71578500 Ki = 0.53 nM T16987 CZ1R3F 71578570 Ki = 2.3 nM T16987 CV0G1A 71578571 Ki = 2.4 nM T16987 CX7T2V 71578640 Ki = 0.64 nM T16987 CVTN91 71578980 Ki = 73.9 nM T16987 CBJ18U 71578981 Ki = 1277 nM T16987 CCKJ51 71578982 Ki = 39.7 nM T16987 C0TKR8 71579053 Ki = 96 nM T16987 CX4D6V 71579054 Ki = 1521 nM T16987 CJ0UP9 71579055 Ki = 79.4 nM T16987 CREN23 71579056 Ki = 1947 nM T16987 CP61GE 71579057 Ki = 1145 nM T16987 CXD68U 71579058 Ki = 79.8 nM T16987 C19OIY 71579130 Ki = 780 nM T16987 CV0LU6 71602117 Ki = 500 nM T16987 CCE15B 71602410 Ki = 0.68 nM T16987 CCB72P 71602411 Ki = 0.6 nM T16987 CHL16T 71602412 Ki = 0.85 nM T16987 C2UQV5 71602471 Ki = 3.1 nM T16987 C8K1YM 71602472 Ki = 2.7 nM T16987 CZL96Y 71602476 Ki = 0.69 nM T16987 CE70AQ 71602537 Ki = 119 nM T16987 C3KPA8 71602538 Ki = 1 nM T16987 CO6FJ4 71602539 Ki = 0.93 nM T16987 CQ17LM 71602540 Ki = 1.1 nM T16987 C1OPS4 71658869 Ki = 1520 nM T16987 CN2FZ3 71659103 Ki = 47 nM T16987 CC0EU9 71677604 Ki = 45.9 nM T16987 CS4VW3 71681364 Ki = 74.7 nM T16987 C5SY2L 71681517 Ki = 622 nM T16987 CT1D0W 71681519 Ki = 705 nM T16987 CW65GP 71681521 Ki = 744 nM T16987 CFS62D 71681523 Ki = 63.3 nM T16987 C96OCT 71681525 Ki = 3.6 nM T16987 C57BRD 71681527 Ki = 750 nM T16987 CU45ER 71681529 Ki = 737 nM T16987 C7NMJ2 71714066 Ki = 24500 nM T16987 C5DEF6 71714067 Ki = 10800 nM T16987 C50LSJ 71714068 Ki = 1480 nM T16987 C84WSV 71716939 Ki = 219 nM T16987 CBY8J3 71716994 Ki = 1100 nM T16987 CM4T1R 71717003 Ki = 1790 nM T16987 CI0SY3 71717570 Ki = 234 nM T16987 CYGT30 71717571 Ki = 254 nM T16987 CG4I1X 71718239 Ki = 400 nM T16987 CVHT94 71718249 Ki = 1 nM T16987 C4N3VH 71718790 Ki = 2.699 nM T16987 CP5J4A 71718856 Ki = 0.98 nM T16987 C0LYX1 71718858 Ki = 890 nM T16987 C7U6NR 71719377 Ki = 717 nM T16987 CM24ND 71719433 Ki = 880 nM T16987 CT3D5S 71719441 Ki = 730 nM T16987 CJG34A 71720036 Ki = 770 nM T16987 CIU4L2 71720670 Ki = 760 nM T16987 CN0L8Q 71720672 Ki = 298 nM T16987 CY54DH 71728127 Ki > 10000 nM T16987 C9JAE7 71728128 Ki > 10000 nM T16987 C6HOP3 71728129 Ki > 10000 nM T16987 CRY5D8 71728130 Ki > 10000 nM T16987 CM91JE 71728236 Ki > 10000 nM T16987 C30ZEI 71728237 Ki > 10000 nM T16987 C4JB8W 71728238 Ki > 10000 nM T16987 C5RS9P 71728239 Ki > 10000 nM T16987 CRYC54 71728240 Ki > 10000 nM T16987 C5TKY7 71764398 Ki = 2.1 nM T16987 CMD91U 71764399 Ki = 6.3 nM T16987 CXO1T9 71764400 Ki = 4.2 nM T16987 CVEI80 71764401 Ki = 0.62 nM T16987 CVQ1H3 71764402 Ki = 1.8 nM T16987 CRZ64M 71764403 Ki = 6.6 nM T16987 CC0X1H 71764607 Ki = 3.1 nM T16987 CK7NI0 71764608 Ki = 1.3 nM T16987 C90YMG 71764609 Ki = 0.24 nM T16987 CK35HL 71764610 Ki = 4.8 nM T16987 C4SV1I 71764611 Ki = 2.3 nM T16987 C8NG9B 71764612 Ki = 0.91 nM T16987 CA2M1B 71764613 Ki = 0.54 nM T16987 CR7J6M 71764825 Ki = 1.5 nM T16987 CG09CJ 71764826 Ki = 0.83 nM T16987 CK2N0Z 71764827 Ki = 3.4 nM T16987 C08RAW 71765040 Ki = 2.5 nM T16987 CGI1J3 71765041 Ki = 0.74 nM T16987 CPT1X2 71765042 Ki = 0.63 nM T16987 CGA62Y 71770789 Ki = 7.3 nM T16987 C8GP3J 71770790 Ki = 6.2 nM T16987 C04WFV 71770791 Ki = 8.8 nM T16987 CN4QC0 71770911 Ki = 45.4 nM T16987 C6XSA1 71770912 Ki = 8.4 nM T16987 C5YU4I 71770913 Ki = 7.4 nM T16987 C4G3HO 71770914 Ki = 107.5 nM T16987 CSU93P 71770915 Ki = 30.3 nM T16987 C9NAK1 71770916 Ki = 6 nM T16987 C42KOE 71770917 Ki = 24.7 nM T16987 CE8IC7 71770918 Ki = 6.6 nM T16987 CQJI19 71771031 Ki = 58.8 nM T16987 C2ZOB7 71771032 Ki = 9.6 nM T16987 C93LEJ 71771033 Ki = 3.4 nM T16987 C5UZM3 71771034 Ki = 239 nM T16987 CX9N5F 71818212 Ki = 293.7 nM T16987 C5IU0Y 72163201 Ki = 6.1 nM T16987 C0Q5XL 72163343 Ki = 12.3 nM T16987 C63MIX 72163344 Ki = 10.2 nM T16987 CL3WV2 72163345 Ki = 19 nM T16987 C4T9DA 72163346 Ki = 197 nM T16987 CTK07O 72163347 Ki = 7.5 nM T16987 CE32BF 72163348 Ki = 5.9 nM T16987 CA1X6Z 72163476 Ki = 6.5 nM T16987 C0FM1E 72202020 Ki = 21 nM T16987 CT41SJ 72202021 Ki = 416 nM T16987 C7WDI2 72204321 Ki = 62.02 nM T16987 CX4G0R 72204928 IC50 = 269 nM T16987 CG9C6U 72204929 IC50 = 239 nM T16987 C5A6XZ 72204930 IC50 = 419 nM T16987 C0XZK4 72204931 IC50 = 89 nM T16987 C6RY4X 72204933 IC50 = 78 nM T16987 C4N5AB 72204934 IC50 = 92 nM T16987 C3H2FZ 72205111 IC50 = 8687 nM T16987 CQ0VX7 72205112 IC50 > 10000 nM T16987 CQ7TI1 72205113 IC50 > 10000 nM T16987 CPAW52 72205114 IC50 > 10000 nM T16987 C2LD3J 72205115 IC50 > 10000 nM T16987 C4E2VS 72543811 Ki = 629 nM T16987 C3UJ8A 72695827 Ki = 40 nM T16987 CX82JD 72696463 Ki = 10 nM T16987 COCV73 72696591 Ki = 4.6 nM T16987 C5KHD7 72696592 Ki = 17.5 nM T16987 C4FBA6 72696593 Ki = 15.4 nM T16987 CO1JM5 72696594 Ki = 5 nM T16987 CUF61Q 72696595 Ki = 4.5 nM T16987 C1SU0Q 72712917 Ki = 8.9 nM T16987 COD5F4 72712918 Ki = 38 nM T16987 CJW7K4 72712919 Ki > 20000 nM T16987 CT2J8A 72712920 Ki > 20000 nM T16987 CRGC51 72713105 Ki = 37 nM T16987 C61VGR 72713106 Ki = 8 nM T16987 C96WHB 72713107 Ki = 8.5 nM T16987 CHPN94 72713108 Ki = 7.6 nM T16987 CJB8R7 72792832 Ki = 7.4 nM T16987 C5F7DT 72792833 Ki = 50.2 nM T16987 CAC7J8 72792834 Ki = 52.7 nM T16987 CFS02B 72792835 Ki = 52 nM T16987 CF5LW1 72792901 Ki = 85.4 nM T16987 C42IFJ 72792902 Ki = 55.1 nM T16987 CRMF25 72792903 Ki = 73.2 nM T16987 C2G5SR 72792904 Ki = 71.9 nM T16987 C6DR9O 72792905 Ki = 44.1 nM T16987 CGF5O1 72792967 Ki = 61.4 nM T16987 CWH3N9 72792968 Ki = 5.4 nM T16987 C5DSF8 72792969 Ki = 9.5 nM T16987 C2K6UZ 72792970 Ki = 31 nM T16987 CGI8K5 72793036 Ki = 23.3 nM T16987 C8WO6Z 72793037 Ki = 35 nM T16987 C6OZ0L 72793038 Ki = 61.9 nM T16987 CDTQ64 72793039 Ki = 53.3 nM T16987 CY16FM 72793040 Ki = 61.1 nM T16987 CXQN80 72793101 Ki = 43.2 nM T16987 CJ19BH 72793102 Ki = 31.4 nM T16987 CO1JT3 73054728 Ki = 6.8 nM T16987 C4MIP9 73345840 Ki = 745 nM T16987 C4Z7PY 73346473 Ki = 29.9 nM T16987 C48AKL 73346474 Ki = 293 nM T16987 CY2AH8 73346475 Ki = 34.8 nM T16987 C8QJU7 73346691 Ki = 7.4 nM T16987 C0PA8K 73346692 Ki = 5.9 nM T16987 CT6C3G 73346693 Ki = 11 nM T16987 CVN4A3 73346695 Ki = 30 nM T16987 CM9K3D 73346697 Ki = 27 nM T16987 C3Y4VZ 73347324 Ki = 0.77 nM T16987 C1WQ0C 73347968 Ki = 76.2 nM T16987 CEHI16 73348197 Ki = 12 nM T16987 C18GUI 73348198 Ki > 1000 nM T16987 C3CJ0F 73349055 Ki > 10000 nM T16987 C75IEZ 73349056 Ki > 10000 nM T16987 CK7MD1 73349516 Ki = 22.6 nM T16987 CJRE74 73349517 Ki = 16.8 nM T16987 CK98JL 73349518 Ki = 569 nM T16987 C6S7RY 73349758 Ki = 17 nM T16987 C2JP5U 73349759 Ki = 4.54 nM T16987 CBL42E 73350409 Ki = 4.1 nM T16987 CP3E7Q 73350410 Ki = 0.78 nM T16987 C38QDY 73351066 Ki = 34.2 nM T16987 COM17Y 73351067 Ki = 326 nM T16987 CN96PE 73351280 Ki = 8.5 nM T16987 CX1J7D 73352124 Ki > 10000 nM T16987 CXJL10 73352125 Ki > 10000 nM T16987 CBN25I 73352538 Ki = 55.3 nM T16987 CRDB68 73352539 Ki = 554 nM T16987 C4SNT8 73352540 Ki = 768 nM T16987 C3M2UH 73354029 Ki = 165 nM T16987 CB7Z2K 73355560 Ki = 27.8 nM T16987 CR81ON 73355561 Ki = 39.1 nM T16987 C60FZE 73355562 Ki = 475 nM T16987 CAK9J2 73355834 Ki = 29 nM T16987 CC2P6U 73356651 Ki > 10000 nM T16987 CC9AE6 73356652 Ki > 10000 nM T16987 C3SB2W 73357104 Ki = 413 nM T16987 C79KVE 73357105 Ki = 87.1 nM T16987 COP7H8 73357339 Ki = 15 nM T16987 CA3YT9 73894059 Ki = 3.9 nM T16987 C53JCV 74766009 Ki = 0.79 nM T16987 C53PBO 74766010 Ki = 0.67 nM T16987 CLPY57 74766011 Ki = 9.6 nM T16987 C7EF5V 76310135 Ki = 68 nM T16987 CLX6H0 76310136 Ki = 54 nM T16987 C9K6XP 76310137 Ki = 28 nM T16987 CX0Y6K 76310141 Ki = 451 nM T16987 C54AJY 76310148 Ki = 0.96 nM T16987 CCD80R 76310490 Ki = 6.3 nM T16987 CUB9V2 76310833 Ki = 63 nM T16987 C4S3QC 76310834 Ki = 18 nM T16987 CY7AV1 76310835 Ki = 10.4 nM T16987 CTJ50C 76310908 Ki = 970 nM T16987 CEWJ18 76310909 Ki = 240 nM T16987 CR9G4Q 76311013 Ki = 17.1 nM T16987 CE7O5U 76311014 Ki = 18.9 nM T16987 CV19YL 76311015 Ki = 10.6 nM T16987 CO0PZ4 76311101 Ki = 17.7 nM T16987 CGT0J3 76311102 Ki = 7.6 nM T16987 CG2JI0 76313836 Ki = 26 nM T16987 CD1A5Y 76313837 Ki = 8.1 nM T16987 CU48XE 76313838 Ki = 40 nM T16987 C04EFJ 76313840 Ki = 134 nM T16987 CZ60NF 76313841 Ki = 429 nM T16987 C5S3XY 76313842 Ki = 540 nM T16987 CK2LR8 76313848 Ki = 6.1 nM T16987 CI3WQ5 76313849 Ki = 5 nM T16987 C0KVD7 76314143 Ki = 7.1 nM T16987 CE1H8W 76314144 Ki = 4.3 nM T16987 C5EM0L 76314145 Ki = 5.7 nM T16987 C0T8HW 76314452 Ki = 24 nM T16987 CZ0JC7 76314453 Ki = 9.5 nM T16987 CC1Z6A 76314549 Ki = 1310 nM T16987 CA1F9S 76314550 Ki > 50000 nM T16987 CZBG52 76314647 Ki = 3.9 nM T16987 C4F7WP 76314648 Ki = 43.7 nM T16987 C95DKS 76314709 Ki = 6.3 nM T16987 C37XBL 76314710 Ki = 5.5 nM T16987 C2H7ZA 76314711 Ki = 44 nM T16987 C34MRW 76317361 Ki = 320 nM T16987 CXZU92 76317371 Ki = 11 nM T16987 CB1VD3 76317966 Ki = 18.5 nM T16987 C6GOE1 76318042 Ki = 4.9 nM T16987 CGQ67N 76318218 Ki = 8.9 nM T16987 CLC1H8 76318279 Ki = 5.9 nM T16987 CT7G2Z 76318280 Ki = 5.5 nM T16987 CCO80M 76318281 Ki = 9.2 nM T16987 CY5O9B 76318282 Ki = 8.9 nM T16987 CM5IV7 76318283 Ki = 30.1 nM T16987 C4DMY8 76318284 Ki = 7.2 nM T16987 CG8QV5 76318285 Ki = 31.2 nM T16987 CDGH94 76321081 Ki = 38 nM T16987 CQ5B4S 76321082 Ki = 46 nM T16987 C9U3LR 76321089 Ki = 442 nM T16987 CZ2RY8 76321096 Ki = 19 nM T16987 C82NGW 76321408 Ki > 10000 nM T16987 CWM9C3 76321409 Ki = 96 nM T16987 C78KRT 76321425 Ki = 6.1 nM T16987 CJ20ZB 76321688 Ki = 4.1 nM T16987 CVT3O8 76321689 Ki = 8.6 nM T16987 CH36SX 76321755 Ki = 45 nM T16987 C8SZN7 76321756 Ki = 56 nM T16987 CP24WC 76321814 Ki = 240 nM T16987 CNP1B7 76321907 Ki = 10.4 nM T16987 C4YP7A 76321908 Ki = 24.3 nM T16987 CZ98LC 76324732 Ki = 6.4 nM T16987 CW87DO 76324733 Ki = 50 nM T16987 C5JXE8 76324738 Ki = 98 nM T16987 CUG2O8 76324739 Ki = 319 nM T16987 CLN0I8 76325020 Ki = 8.1 nM T16987 C35EUT 76325021 Ki = 5.4 nM T16987 CZQ93S 76325300 Ki = 15.1 nM T16987 CP3X6L 76325374 Ki = 4.5 nM T16987 CO79TZ 76325375 Ki = 12.7 nM T16987 CE1DM0 76325376 Ki = 4.9 nM T16987 CE3P4W 76325377 Ki = 8.9 nM T16987 C7ZJ9M 76325378 Ki = 3.6 nM T16987 CN6CY7 76325452 Ki = 250 nM T16987 CUC3M2 76325547 Ki = 10.2 nM T16987 C1BC4A 76325548 Ki = 12.9 nM T16987 CQUE95 76325602 Ki = 6.9 nM T16987 CDO73V 76325603 Ki = 42.9 nM T16987 C0UK2H 76328279 Ki = 43 nM T16987 CCNB68 76328280 Ki = 218 nM T16987 C8AS9R 76328281 Ki = 28 nM T16987 C0CFZ1 76328574 Ki = 491 nM T16987 CYM2G9 76328575 Ki = 838 nM T16987 CZ5X4W 76328576 Ki = 620 nM T16987 CP3CN4 76328593 Ki = 8.8 nM T16987 CPJM79 76328853 Ki = 12.3 nM T16987 C6F4LU 76328915 Ki = 18 nM T16987 C5VW9J 76328916 Ki = 20 nM T16987 CEZ6A8 76328917 Ki = 43 nM T16987 CYD50A 76329098 Ki = 13 nM T16987 CB23PR 76329099 Ki = 23 nM T16987 C3QI6J 76329100 Ki = 10.7 nM T16987 CTF2G1 76329169 Ki = 7.6 nM T16987 CAE23D 76329170 Ki = 7.8 nM T16987 CKH0X7 76331969 Ki = 40 nM T16987 CO82ZX 76331970 Ki = 39 nM T16987 C5U7JI 76331976 Ki = 523 nM T16987 CYC39A 76331984 Ki = 18 nM T16987 CK73VH 76331985 Ki = 63 nM T16987 C68DOK 76332270 Ki = 6.4 nM T16987 CJN0W8 76332271 Ki = 59.8 nM T16987 C3ZGF1 76332272 Ki = 13.5 nM T16987 C6ENW5 76332521 Ki = 4.3 nM T16987 C4RPU5 76332522 Ki = 2.1 nM T16987 C14UQS 76332523 Ki = 25.4 nM T16987 CGLB34 76332602 Ki = 3 nM T16987 CP9SU7 76332603 Ki = 21 nM T16987 CG3U6D 76332757 Ki = 13.5 nM T16987 CSN84K 76332758 Ki = 1.9 nM T16987 COZ89H 76332830 Ki = 5.7 nM T16987 CFI5K7 76332831 Ki = 9.2 nM T16987 C5VN9Q 76332832 Ki = 9.5 nM T16987 C9W0HZ 76335546 Ki = 84 nM T16987 CZC97G 76335551 Ki = 340 nM T16987 CQKW51 76335889 Ki = 3746 nM T16987 CB53XC 76335911 Ki = 7.3 nM T16987 CP16NU 76336199 Ki = 3.8 nM T16987 C3P4ZB 76336200 Ki = 1.3 nM T16987 CLB17E 76336381 Ki = 21.5 nM T16987 CV1B6C 76336382 Ki = 4.5 nM T16987 CWFY73 76336452 Ki = 6.7 nM T16987 C2QC4D 76336453 Ki = 9.4 nM T16987 CH0OY6 78319159 Ki = 9 nM T16987 CC4F0A 78319160 Ki = 7.1 nM T16987 CO4IE9 78319161 Ki = 7.5 nM T16987 CY6LN4 78319162 Ki = 7.9 nM T16987 CU9I6V 82078731 Ki = 42.7 nM T16987 C5TB6O 82080973 Ki = 38.3 nM T16987 CX5WB9 82198349 Ki = 3.2 nM T16987 C6UZR9 82911195 Ki = 2.3 nM T16987 CVD64Q 83379931 Ki = 125 nM T16987 CR47YB 86047482 Ki = 7.1 nM T16987 C0P3OF 86047486 Ki = 6.5 nM T16987 CZ5HA6 86047495 Ki = 8.3 nM T16987 CTD2Y9 86276273 Ki = 12 nM T16987 CHY2O4 86276274 Ki = 12 nM T16987 CN7HU3 86288843 Ki = 5.9 nM T16987 C5Y1WO 86288855 Ki = 5.7 nM T16987 C76RBA 86298624 IC50 = 87 nM T16987 C93FKI 86298625 IC50 = 76 nM T16987 CVLU48 86298626 IC50 = 65 nM T16987 CR97VD 86692717 Ki = 6.6 nM T16987 C8PC3U 86692718 Ki = 6.4 nM T16987 C6HC8V 86692720 Ki = 9.1 nM T16987 CQ30FJ 86719933 Ki = 27 nM T16987 CH2X9D 88314331 Ki = 37.8 nM T16987 C3EYT4 88314336 Ki = 4.8 nM T16987 C1O5YX 90180909 Ki = 410 nM T16987 CIJ96H 90644155 IC50 = 62 nM T16987 CX7EW1 90644156 IC50 = 278 nM T16987 CK5GZ4 90644157 IC50 = 225 nM T16987 C7O1YN 90644158 IC50 = 376 nM T16987 CEN6C1 90644159 IC50 = 92 nM T16987 C8X9UZ 90644160 IC50 = 794 nM T16987 C4QT6W 90644479 Ki = 3.6 nM T16987 C6XB9R 90644480 Ki = 23 nM T16987 C1KXA0 90644481 Ki = 33 nM T16987 C1ND2E 90644482 Ki = 24 nM T16987 CY4LZ9 90644483 Ki = 32 nM T16987 C2RQD9 90644484 Ki = 44 nM T16987 CZ0R6T 90644485 Ki = 95 nM T16987 C4G1BD 90644486 Ki = 24 nM T16987 CL7I9M 90644487 Ki = 30 nM T16987 CVMU79 90644488 Ki = 8.4 nM T16987 C6F5ZP 90644489 Ki = 4.7 nM T16987 CG85NB 90644490 Ki = 5 nM T16987 CCID31 90644491 Ki = 2.7 nM T16987 C3BPF8 90644492 Ki = 8.1 nM T16987 C7B5YR 90644493 Ki = 7.6 nM T16987 C9FCX5 90644494 Ki = 6.3 nM T16987 CQND72 90644495 Ki = 12.5 nM T16987 C4V9IZ 90644496 Ki = 8.9 nM T16987 C49VLZ 90644497 Ki = 7.1 nM T16987 CX2I9G 90644498 Ki = 6.4 nM T16987 C5MXJ4 90644499 Ki = 8 nM T16987 C2E7QM 90644500 Ki = 13.6 nM T16987 CR02MV 90644501 Ki = 8.2 nM T16987 C2SZ5P 90644502 Ki = 5.4 nM T16987 C86NMC 90644503 Ki = 2.8 nM T16987 C8W3PI 90644504 Ki = 4.3 nM T16987 CF12MK 90645415 Ki = 0.74 nM T16987 CJO6I7 90645416 Ki = 31.6 nM T16987 CU2K5R 90645417 Ki = 211 nM T16987 C58KIU 90645418 Ki = 70.8 nM T16987 CS0OX7 90645419 Ki = 365 nM T16987 CWD6P7 90645420 Ki = 184 nM T16987 CVY5P9 90645421 Ki = 79.2 nM T16987 CAL9C4 90645422 Ki = 9.3 nM T16987 C2EA9C 90645423 Ki = 9.2 nM T16987 C1FVA8 90645424 Ki = 0.76 nM T16987 CP27AX 90645425 Ki = 0.912 nM T16987 C8E4ZH 90645426 Ki = 5.4 nM T16987 C3SIA9 90645429 Ki = 0.72 nM T16987 C1E4FS 90645430 Ki = 0.81 nM T16987 COBQ09 90645431 Ki = 0.94 nM T16987 C7IU8K 90645432 Ki = 3.4 nM T16987 CW0L1D 90654798 Ki = 6.2 nM T16987 CO2CU1 90654800 Ki = 6.2 nM T16987 CE54MK 90654802 Ki = 5.3 nM T16987 CID9U2 90654804 Ki = 8.1 nM T16987 C27QHW 90654822 Ki = 665 nM T16987 C96OWE 90654823 Ki = 86.2 nM T16987 CZQ9E3 90654824 Ki = 57.3 nM T16987 CCPO43 90654825 Ki = 747 nM T16987 C4D2TM 90654826 Ki = 866 nM T16987 C48XBN 90654827 Ki = 81.2 nM T16987 CI8TG3 90654828 Ki = 201 nM T16987 C6GFZ0 90654829 Ki = 9.5 nM T16987 C3Z1GS 90654830 Ki = 572 nM T16987 C4JSW5 90655322 Ki = 38 nM T16987 C3QH0R 90655323 Ki = 21 nM T16987 CF0U7K 90655324 Ki = 35 nM T16987 CU31VY 90675933 Ki = 636 nM T16987 C2XWG7 90675934 Ki = 616 nM T16987 CH7R2B 90675935 Ki = 30.2 nM T16987 CORQ94 90675936 Ki = 579 nM T16987 CE39DC 90675937 Ki = 606 nM T16987 CSU5K2 90675938 Ki = 667 nM T16987 CE8S1J 90675939 Ki = 57.3 nM T16987 C1H9FB 90675940 Ki = 59.5 nM T16987 CPB36R 90675941 Ki = 7.3 nM T16987 C28FLQ 91498333 Ki = 745 nM T16987 CE6LO5 91595667 Ki = 8.5 nM T16987 C3AYZ5 91811067 Ki = 27 nM T16987 CE2OY1 91995964 Ki = 25.4 nM T16987 CX45AP 92044053 Ki = 4.1 nM T16987 CEH68Q 93972064 Ki = 9.7 nM T16987 CE8GH2 101874826 Ki = 5.9 nM T16987 C4W9FG 101874827 Ki = 6.4 nM T16987 CY7G8A 101874828 Ki = 5.1 nM T16987 C1TM8I 101874829 Ki = 5.6 nM T16987 CVZ3L5 101874830 Ki = 6.8 nM T16987 C2H5FC 101876957 Ki = 4.5 nM T16987 CDGZ03 101879106 Ki = 6.2 nM T16987 CY6ER7 101879108 Ki = 43 nM T16987 CAC1W7 101913750 Ki = 80 nM T16987 CQX8K1 101913751 Ki = 682 nM T16987 CIP25Q 101913752 Ki = 653 nM T16987 CTY15S 101913753 Ki = 236 nM T16987 C49NEJ 101913754 Ki = 89 nM T16987 CW5Q7L 101913755 Ki = 84 nM T16987 CE90SD 102138248 Ki = 15.3 nM T16987 CP1X9Y 102232756 Ki = 500 nM T16987 CQBE51 102341119 Ki = 1 nM T16987 C2TX7A 102354117 Ki = 14.2 nM T16987 CK43QR 102405972 Ki = 126 nM T16987 C6LUE5 109059506 Ki = 398 nM T16987 CUY64D 109061586 Ki = 34.7 nM T16987 CXN7Z8 110453853 Ki = 20.3 nM T16987 C6I0LD 112499923 Ki = 4.3 nM T16987 C8CFR6 112499924 Ki = 0.58 nM T16987 CUR4V8 114816322 Ki = 4.7 nM T16987 C3TZ9A 115950959 Ki = 131 nM T16987 CAO67C 118705769 Ki = 26.4 nM T16987 CW1D8A 118705770 Ki = 6.6 nM T16987 CTFB51 118705771 Ki = 23.7 nM T16987 C5NGT8 118705772 Ki = 7.1 nM T16987 C3G4ZN 118705773 Ki = 7.9 nM T16987 CBVD13 118705774 Ki = 6.3 nM T16987 C3KCZ6 118705775 Ki = 77.8 nM T16987 C5Z4QF 118705776 Ki = 82.3 nM T16987 CV4YN0 118705777 Ki = 6.1 nM T16987 C0IBQ8 118705778 Ki = 6.3 nM T16987 CH7LV5 118705779 Ki = 3.9 nM T16987 CU5SI9 118705780 Ki = 3.8 nM T16987 C6IGP0 118705781 Ki = 6.2 nM T16987 C7ZE2H 118705782 Ki = 6 nM T16987 C47QFN 118705783 Ki = 70.3 nM T16987 CO1P3T 118705784 Ki = 72.5 nM T16987 CK8E5C 118705785 Ki = 28.4 nM T16987 CS9G2U 118705786 Ki = 30.1 nM T16987 C1XV9M 118705787 Ki = 5.6 nM T16987 C7GW3Q 118705788 Ki = 5.9 nM T16987 CUIS94 118706141 Ki = 3.1 nM T16987 CET19U 118706142 Ki = 2.9 nM T16987 C6FBG3 118706893 Ki = 42.5 nM T16987 C1CLV5 118706959 Ki = 410 nM T16987 CLA5I2 118706960 Ki = 201 nM T16987 C8GD4Y 118706961 Ki = 352 nM T16987 CB0E4N 118706962 Ki = 407 nM T16987 CPI7L3 118710135 Ki = 103 nM T16987 C05ZCN 118710136 Ki = 85.8 nM T16987 C45XHE 118710137 Ki = 178 nM T16987 C84YKV 118710138 Ki = 2900 nM T16987 CFA76H 118710139 Ki = 159 nM T16987 C0UWK2 118710140 Ki = 157 nM T16987 CGJ59E 118710141 Ki = 4530 nM T16987 C64BUR 118710142 Ki = 2710 nM T16987 C1W2DB 118710143 Ki = 2170 nM T16987 CZ4F3O 118710144 Ki = 2830 nM T16987 CWR82N 118710145 Ki = 177 nM T16987 C7R5FO 118710146 Ki = 134 nM T16987 CD8U1O 118710147 Ki = 180 nM T16987 C8YFH6 118710148 Ki = 170 nM T16987 CLPC68 118710149 Ki = 180 nM T16987 C8OH4V 118710150 Ki = 18.3 nM T16987 C6CAQ4 118710151 Ki = 91.5 nM T16987 CS0G7T 118710152 Ki = 170 nM T16987 C3NPF1 118710200 Ki = 136 nM T16987 C4YXF1 118710201 Ki = 16.5 nM T16987 C1B5QL 118710202 Ki = 126 nM T16987 CUJ42P 118710203 Ki = 16.3 nM T16987 CK23DF 118710598 Ki = 0.68 nM T16987 CS9MC2 118710599 Ki = 0.72 nM T16987 CW2D4O 118710600 Ki = 0.63 nM T16987 CTMF04 118710601 Ki = 0.79 nM T16987 CU2C9L 118710602 Ki = 0.65 nM T16987 CFCG50 118710603 Ki = 0.79 nM T16987 C2G5DI 118710604 Ki = 0.59 nM T16987 CY2S9V 118710605 Ki = 0.66 nM T16987 C5L6IK 118710606 Ki = 0.71 nM T16987 C6ZGB2 118711612 Ki = 1.4 nM T16987 CNS6L8 118711613 Ki = 12.4 nM T16987 CY0E8G 118711614 Ki = 2.5 nM T16987 CI71PW 118711615 Ki = 2.3 nM T16987 C1X7RI 118711616 Ki = 2 nM T16987 C7P6GM 118711617 Ki = 62.6 nM T16987 CYNA84 118711618 Ki = 1.9 nM T16987 CL38UN 118711619 Ki = 1.9 nM T16987 CGUV98 118711620 Ki = 5.7 nM T16987 CJ2UH6 118711621 Ki = 10.8 nM T16987 CH2RE7 118711622 Ki = 0.8 nM T16987 C1RWN4 118711623 Ki = 0.9 nM T16987 CR0I6S 118711624 Ki = 1.1 nM T16987 C8LQI3 118711625 Ki = 2.6 nM T16987 C5SEJ6 118711626 Ki = 3.6 nM T16987 C5TYE7 118711627 Ki = 2.7 nM T16987 C7ZOH6 118712658 Ki = 794 nM T16987 C19IXJ 118712659 Ki = 589 nM T16987 CD5MB4 118712660 Ki = 81 nM T16987 C0EPI8 118712661 Ki = 235 nM T16987 CZ18GD 118716360 Ki = 9 nM T16987 CX6F4B 118716361 Ki = 94 nM T16987 CO4K8Z 118716362 Ki = 9 nM T16987 CR8HX4 118716363 Ki = 60 nM T16987 CYH2P1 118716364 Ki = 8 nM T16987 C61BOY 118716365 Ki = 85 nM T16987 C8PJC3 118716366 Ki = 1 nM T16987 C9HP7J 118716367 Ki = 21 nM T16987 CTS52R 118716368 Ki = 85 nM T16987 CHI60Z 118716369 Ki = 34 nM T16987 CA1UY4 118716496 Ki = 19.3 nM T16987 CVR32C 118716497 Ki = 5.6 nM T16987 CT1RQ6 118716498 Ki = 5.4 nM T16987 CG10AC 118716499 Ki = 0.96 nM T16987 CV89MK 118716500 Ki = 0.95 nM T16987 C57YMW 118716501 Ki = 0.81 nM T16987 CQ73KL 118716502 Ki = 0.67 nM T16987 CXE59K 118716504 Ki = 0.68 nM T16987 CONM87 118716505 Ki = 79.3 nM T16987 CQ3I7N 118716509 Ki = 28.6 nM T16987 C72KER 118716510 Ki = 9.1 nM T16987 C0RJI1 118716511 Ki = 8.6 nM T16987 CFU0Z8 118716512 Ki = 9.5 nM T16987 CXU4D7 118716513 Ki = 8.3 nM T16987 C86KQZ 118716514 Ki = 15 nM T16987 C9HLA8 118716891 Ki = 76 nM T16987 CJ0YC9 118716892 Ki = 207 nM T16987 CJ8TZ3 118716893 Ki = 86 nM T16987 C0X1WQ 118716894 Ki = 81 nM T16987 CDG4L8 118716895 Ki = 93 nM T16987 CFD26B 118716950 Ki = 617 nM T16987 C20YBM 118716951 Ki = 614 nM T16987 C0V1ZT 118716952 Ki = 58 nM T16987 CH9BW0 118716953 Ki = 349 nM T16987 CXB89Y 118716954 Ki = 611 nM T16987 C8CKU2 118716955 Ki = 307 nM T16987 CF03IX 118716956 Ki = 54.4 nM T16987 CYN29C 118716960 Ki = 35.5 nM T16987 C4AC7H 118716961 Ki = 241 nM T16987 CJ9O3I 118716962 Ki = 123 nM T16987 C6RJ9W 118716964 Ki = 12.9 nM T16987 CMVW90 118716999 Ki = 93 nM T16987 CBKN39 118717000 Ki = 68 nM T16987 C6N8CF 118717001 Ki = 88 nM T16987 CL3P7I 118717002 Ki = 415 nM T16987 C2H0NP 118717003 Ki = 87 nM T16987 CXRD23 118719969 Ki = 4.1 nM T16987 C4Z6DI 118719970 Ki = 4.6 nM T16987 C2HJ4Y 118719971 Ki = 68.5 nM T16987 CD1OH8 118719972 Ki = 9.4 nM T16987 C0R8JN 118719973 Ki = 8.9 nM T16987 CMR0H2 118719974 Ki = 6 nM T16987 CI3QG5 118719975 Ki = 7.7 nM T16987 C06YTV 118719976 Ki = 7.6 nM T16987 C25BJT 118721385 Ki = 214 nM T16987 CI4W0E 118721386 Ki = 264 nM T16987 CFRX59 118721387 Ki = 172 nM T16987 C5SYD7 118721388 Ki > 10000 nM T16987 CNT18B 118721389 Ki = 39.8 nM T16987 CYC50E 118721390 Ki = 74.5 nM T16987 CYL0W1 118721391 Ki = 38.7 nM T16987 C1HN6R 118721392 Ki = 53.5 nM T16987 C2WLI4 118721393 Ki = 65.2 nM T16987 CQVS30 118721394 Ki = 29.9 nM T16987 CL2Q8M 118721395 Ki = 5.5 nM T16987 CAG5L6 118721396 Ki = 97.4 nM T16987 CJ63BR 118721397 Ki = 6.6 nM T16987 C14ZNT 118721398 Ki = 7.2 nM T16987 C1J6IX 118721399 Ki = 20.3 nM T16987 CVJ92D 118721400 Ki = 7.4 nM T16987 C5F7PT 118721401 Ki = 284 nM T16987 C5AFR3 118721402 Ki = 30.2 nM T16987 C29EYL 118721403 Ki = 34.9 nM T16987 C8GYO9 118721404 Ki = 48.2 nM T16987 CSZ7Q0 118721405 Ki = 50.1 nM T16987 CY3ZW6 118721406 Ki = 83.8 nM T16987 C4T9IR 118721407 Ki = 107 nM T16987 CNPB81 118721408 Ki = 96.8 nM T16987 CP40JF 118722001 Ki = 281 nM T16987 CXTR97 118723294 Ki = 7.2 nM T16987 C42JBV 118723295 Ki = 6.5 nM T16987 CVDC56 118723296 Ki = 5.7 nM T16987 C2RG7F 118723303 Ki = 8.6 nM T16987 C0CMO4 118723304 Ki = 5.7 nM T16987 CC7RH0 118723305 Ki = 7.1 nM T16987 CU0R8X 118723306 Ki = 609 nM T16987 C67LPC 118723308 Ki = 36.7 nM T16987 C0D1SQ 118724328 Ki = 37.4 nM T16987 C89YTC 118724329 Ki = 58.3 nM T16987 CBT87C 118724330 Ki = 50.7 nM T16987 C49AWZ 118724331 Ki = 43.5 nM T16987 CP9X5K 118728047 Ki = 9.2 nM T16987 CUA3S7 118728048 Ki = 6.5 nM T16987 C2K3DO 118728049 Ki = 8.3 nM T16987 CZTN86 118728050 Ki = 4.7 nM T16987 C0CUV2 118728051 Ki = 91 nM T16987 CGU5O0 118728053 Ki = 90.1 nM T16987 CGQ69F 118728055 Ki = 93.8 nM T16987 C2JEW0 118728057 Ki = 50.8 nM T16987 CCBJ19 118728058 Ki = 33.3 nM T16987 CKJ8S9 118728060 Ki = 66.2 nM T16987 C0O3BI 118728062 Ki = 24.5 nM T16987 CH2E8F 118728064 Ki = 8.4 nM T16987 C4JM1O 118728066 Ki = 0.76 nM T16987 C67YPT 118728068 Ki = 91.3 nM T16987 CML9F8 118728070 Ki = 8 nM T16987 CA52IR 118728072 Ki = 414 nM T16987 CVE9H5 118728074 Ki = 3.9 nM T16987 CS9ZW3 118728500 Ki = 3.8 nM T16987 CI7MY8 118728501 Ki = 40.9 nM T16987 CZE9K8 118728502 Ki = 608 nM T16987 C8S9JV 118728503 Ki = 5.5 nM T16987 C40AIB 118729374 Ki = 4.9 nM T16987 CO3Z5E 118729375 Ki = 14.2 nM T16987 C6S0DR 118729376 Ki = 5.9 nM T16987 CVXO79 118729377 Ki = 4.6 nM T16987 C62BGK 118729378 Ki = 9.4 nM T16987 C4D9EP 118729379 Ki = 10.5 nM T16987 C2TOH7 118729380 Ki = 8 nM T16987 C5P9ND 118729381 Ki = 3.5 nM T16987 C2XLV4 118729382 Ki = 6.8 nM T16987 CVLK60 118729383 Ki = 3.7 nM T16987 C8U7SE 118729384 Ki = 6.1 nM T16987 CV7OS1 118729385 Ki = 9.1 nM T16987 C7Z2OR 118729386 Ki = 5.7 nM T16987 CHE1K4 118729473 Ki = 0.75 nM T16987 C9V8MA 118729474 Ki = 33.8 nM T16987 C8GJP5 118729475 Ki = 50.4 nM T16987 C4MEZ0 118729476 Ki = 6.2 nM T16987 CE3IV5 118729477 Ki = 4.9 nM T16987 C08EZC 118733945 Ki = 424.04 nM T16987 C3F1DU 118733947 Ki = 79.35 nM T16987 C4OL1A 118733948 Ki = 22.88 nM T16987 CP25HS 118733949 Ki = 10.76 nM T16987 CY3H4E 118736318 Ki = 1045 nM T16987 C8HY4S 118736320 Ki = 1084 nM T16987 C7F5JH 118736322 Ki = 1470 nM T16987 C7MDJ3 118736324 Ki = 85.6 nM T16987 CQM67J 118736325 Ki = 10.5 nM T16987 CKY90W 118736326 Ki = 11.1 nM T16987 CY4B1U 118736327 Ki = 9.5 nM T16987 CRZ1T6 118736328 Ki = 11.3 nM T16987 CFDB97 118737265 Ki = 8.7 nM T16987 CVGF86 118737267 Ki = 3.7 nM T16987 C6B8WR 118737268 Ki = 3.2 nM T16987 CWEM68 118737269 Ki = 8.1 nM T16987 C6PXT8 118737270 Ki = 2.4 nM T16987 CWP7Q1 118737271 Ki = 7 nM T16987 CAB65M 118737272 Ki = 4.8 nM T16987 CHR0I7 118737273 Ki = 4 nM T16987 C72BLG 118737274 Ki = 6.1 nM T16987 C4TD0Q 118737275 Ki = 6.2 nM T16987 CZ1J0U 118737276 Ki = 6.8 nM T16987 CHN09Y 118737277 Ki = 2.1 nM T16987 CMR62B 118737278 Ki = 10.9 nM T16987 C1CV3E 118737279 Ki = 26.6 nM T16987 CP8Y5U 119090745 Ki = 5.6 nM T16987 C4K6CG 119943184 Ki = 851 nM T16987 CHX4Y2 121382833 Ki > 50000 nM T16987 CNEJ87 121382878 Ki = 689 nM T16987 CBHM75 121382881 Ki = 10160 nM T16987 C13GKC 121382882 Ki = 9380 nM T16987 C8QTR4 121382883 Ki = 7340 nM T16987 C96ANJ 121382897 Ki > 50000 nM T16987 CUS64J 121382999 Ki = 12400 nM T16987 C6C4WE 121383002 Ki = 92.7 nM T16987 CG48HD 122164592 Ki = 440 nM T16987 CK92MV 122179845 Ki = 536 nM T16987 C10UQY 122179846 Ki = 77.5 nM T16987 CLV96C 122179847 Ki = 78.1 nM T16987 C2RT1Y 122179848 Ki = 91.5 nM T16987 C06ZSC 122179849 Ki = 82.8 nM T16987 C74RAE 122179850 Ki = 77.8 nM T16987 C6NM0Q 122179851 Ki = 77.6 nM T16987 CYP3B0 122179852 Ki = 70.3 nM T16987 CMP05I 122179853 Ki = 79.4 nM T16987 C2TGN6 122179854 Ki = 81.5 nM T16987 CAH3I1 122179855 Ki = 93.1 nM T16987 C8YJ9B 122180166 Ki = 965 nM T16987 CHON20 122180167 Ki = 256 nM T16987 C9L2TG 122180168 Ki = 419 nM T16987 C9L3OY 122180169 Ki = 66 nM T16987 CJ1X2F 122180170 Ki = 300 nM T16987 CVCX92 122180171 Ki = 9.9 nM T16987 C6LEA3 122180172 Ki = 206 nM T16987 CV8Z4I 122182643 Ki = 9.5 nM T16987 CV96QP 122182644 Ki = 5.8 nM T16987 CA91HP 122182645 Ki = 8.2 nM T16987 C08EBQ 122182646 Ki = 7.7 nM T16987 CSJA24 122182647 Ki = 7.3 nM T16987 CDM51W 122182648 Ki = 9.4 nM T16987 C3E9FK 122182649 Ki = 6.3 nM T16987 CUF5N9 122182650 Ki = 5.7 nM T16987 C5BRH0 122182651 Ki = 6.6 nM T16987 C45DQE 122182654 Ki = 5.2 nM T16987 CDRF43 122182655 Ki = 5.6 nM T16987 CQ83BJ 122182656 Ki = 4.8 nM T16987 CH4Z8B 122182657 Ki = 4.3 nM T16987 CU71LK 122182658 Ki = 4.8 nM T16987 CY1NK4 122182659 Ki = 4.8 nM T16987 CP4I8D 122184891 Ki = 9.4 nM T16987 CZ2RM0 122184892 Ki = 7.1 nM T16987 CFQ4R3 122184893 Ki = 5.9 nM T16987 C69UQF 122184894 Ki = 3 nM T16987 CNF20A 122184895 Ki = 55.7 nM T16987 CJAL95 122184896 Ki = 0.47 nM T16987 C51LFX 122184933 Ki = 0.58 nM T16987 CTQP23 122184934 Ki = 4 nM T16987 CL49QM 122184935 Ki = 0.54 nM T16987 CVN28C 122184936 Ki = 0.57 nM T16987 CU4S6Y 122184937 Ki = 3.9 nM T16987 C4VWG9 122184938 Ki = 5.1 nM T16987 C7H8ZI 122184984 Ki = 1 nM T16987 CX76HF 122184985 Ki = 1 nM T16987 C1KOF6 122184986 Ki = 64.7 nM T16987 C01CWK 122184987 Ki = 84.5 nM T16987 CVTY87 122184988 Ki = 35.8 nM T16987 CM5A7F 122184989 Ki = 1 nM T16987 CYM65N 122184990 Ki = 37 nM T16987 CQ9YU1 122184991 Ki = 1.1 nM T16987 C83GXC 122184992 Ki = 1 nM T16987 CTV40W 122184993 Ki = 1 nM T16987 CWM21G 122184994 Ki = 1 nM T16987 C19LDQ 122184995 Ki = 7.1 nM T16987 C7UE2C 122184996 Ki = 6.3 nM T16987 CWBN52 122184997 Ki = 8.6 nM T16987 C1CI4W 122184998 Ki = 9.5 nM T16987 CWJ94V 122185033 Ki = 9 nM T16987 C9PG8Z 122185234 Ki = 29.5 nM T16987 C93KBM 122185235 Ki = 27.3 nM T16987 CX6Z5Y 122185236 Ki = 6.4 nM T16987 CFPV38 122185237 Ki = 7 nM T16987 CVZ70D 122185238 Ki = 6.7 nM T16987 C14OHP 122185239 Ki = 5.8 nM T16987 CB63WU 122185240 Ki = 5.5 nM T16987 CE3Q1J 122185241 Ki = 8.3 nM T16987 CNG63S 122185242 Ki = 5.3 nM T16987 CY7H0T 122185243 Ki = 6.2 nM T16987 C2ME1I 122185244 Ki = 6.1 nM T16987 C0EPT7 122185245 Ki = 0.46 nM T16987 CI1AL4 122185246 Ki = 6.25 nM T16987 CM43CE 122185684 Ki = 961 nM T16987 CSQ43L 122185685 Ki = 60 nM T16987 CCA9I1 122185686 Ki = 11 nM T16987 CLIR24 122185687 Ki = 8.8 nM T16987 C5NWU9 122185688 Ki = 9.6 nM T16987 CY70TU 122185689 Ki = 8.9 nM T16987 CD94UC 122185690 Ki = 9.1 nM T16987 C8TIP4 122185692 Ki = 277 nM T16987 CE7W6O 122185694 Ki = 52 nM T16987 CV2G7S 122185695 Ki = 11 nM T16987 C1M5JR 122185696 Ki = 742 nM T16987 CMB32C 122185697 Ki = 115 nM T16987 C1FR9Q 122185698 Ki = 101 nM T16987 CY2D9L 122185699 Ki = 49 nM T16987 C2NUJ9 122185700 Ki = 12 nM T16987 CHBC74 122185771 Ki = 78 nM T16987 CZM98F 122185772 Ki = 12 nM T16987 CP8Y5E 122185773 Ki = 12 nM T16987 CK2Q7M 122185774 Ki = 12 nM T16987 CF4L0N 122185776 Ki = 12 nM T16987 C7T4BF 122185778 Ki = 80 nM T16987 C4TZ6G 122185779 Ki = 43 nM T16987 CUI73A 122187162 Ki = 6.2 nM T16987 C1Q7AX 122187163 Ki = 8.7 nM T16987 CO6P7A 122187164 Ki = 42.3 nM T16987 C9LN8Q 122187165 Ki = 6.9 nM T16987 COK6D7 122187166 Ki = 245 nM T16987 C7NV8G 122187167 Ki = 381 nM T16987 C6XKH1 122187168 Ki = 1395 nM T16987 C5KMW2 122187169 Ki = 3535 nM T16987 CSA78D 122187170 Ki = 7960 nM T16987 C5V7SZ 122187171 Ki = 62.8 nM T16987 C6FMG1 122187172 Ki = 2790 nM T16987 CVG1U0 122187173 Ki = 557 nM T16987 CR8NT0 122187174 Ki = 8570 nM T16987 CWSM36 122187175 Ki > 10000 nM T16987 CT59AR 122187176 Ki = 9.4 nM T16987 C93ESN 122187177 Ki = 9.2 nM T16987 CL0JF6 122187178 Ki = 5.1 nM T16987 CQ81UP 122187179 Ki = 6.7 nM T16987 CIE0W8 122187180 Ki = 30.3 nM T16987 CNSU27 122187181 Ki = 3.6 nM T16987 C7LDH1 122187182 Ki = 8.7 nM T16987 CG9T3N 122187183 Ki = 6.6 nM T16987 CBE9U8 122187184 Ki = 64.4 nM T16987 C13USE 122187185 Ki = 9.2 nM T16987 CE36PK 122187423 Ki = 62.5 nM T16987 CDS2I6 122187424 Ki = 46.5 nM T16987 CMF63L 122187425 Ki = 38.1 nM T16987 C7Q9TP 122187426 Ki = 128 nM T16987 C04HSI 122187596 Ki = 49 nM T16987 CZ74KO 122187597 Ki = 556 nM T16987 C07OYV 122187598 Ki = 39 nM T16987 CO6AT2 122187599 Ki = 43 nM T16987 C7WJ4B 122187600 Ki = 43 nM T16987 CZ0Y1G 122187601 Ki = 24 nM T16987 CWF7Z0 122187602 Ki = 24 nM T16987 C07ZNW 122187603 Ki = 58 nM T16987 C7K6TV 122187604 Ki = 80 nM T16987 CX69YT 122187605 Ki = 41 nM T16987 C8XN0F 122187606 Ki = 29 nM T16987 CVT13C 122187607 Ki = 56 nM T16987 CB2DT8 122187638 Ki = 153 nM T16987 C0G4CQ 122187639 Ki = 120 nM T16987 CQSV13 122187640 Ki = 144 nM T16987 CH74EW 122187641 Ki = 247 nM T16987 CH3C8V 122187642 Ki = 17 nM T16987 CP01NQ 122187643 Ki = 17.8 nM T16987 CRM3S4 122188878 Ki = 51.3 nM T16987 C5UF1Q 122188879 Ki = 75.1 nM T16987 CQB9A8 122188880 Ki = 630 nM T16987 C1SFD4 122188881 Ki = 76.8 nM T16987 CIE7L0 122188882 Ki = 90.4 nM T16987 C6MPI4 122189078 Ki = 7.8 nM T16987 C9V7WT 122189088 Ki = 17.7 nM T16987 C1QZV7 122189098 Ki = 9.4 nM T16987 C5XT3S 122192640 Ki = 350 nM T16987 C1LCB9 122192641 Ki = 610 nM T16987 CP51XT 122192642 Ki = 30 nM T16987 C5GKT0 122192643 Ki = 640 nM T16987 C3RZM8 122192644 Ki = 530 nM T16987 CHLG86 122192645 Ki = 920 nM T16987 CTK4J8 122192646 Ki = 860 nM T16987 CVNQ49 122192647 Ki = 260 nM T16987 CX3A0N 122192648 Ki = 370 nM T16987 CU3F1V 122192649 Ki = 1020 nM T16987 CQ4NT8 122192650 Ki = 780 nM T16987 C2REU8 122192651 Ki = 920 nM T16987 CL5P4T 122192652 Ki = 560 nM T16987 C0KF5I 122192653 Ki = 520 nM T16987 CT64DB 122192654 Ki = 830 nM T16987 CX05RY 122192671 Ki = 5.1 nM T16987 CE9ZC4 122192672 Ki = 5.5 nM T16987 CUW2B9 122192673 Ki = 27.1 nM T16987 CKU76Q 122192674 Ki = 5.2 nM T16987 C49KGU 122192675 Ki = 4.7 nM T16987 CB0J2T 122192676 Ki = 5.5 nM T16987 CS63LF 122192677 Ki = 5.3 nM T16987 C4T3IO 122192678 Ki = 4.9 nM T16987 CTZ4L6 122192679 Ki = 9.9 nM T16987 C62VGD 122192680 Ki = 5 nM T16987 CYND20 122192681 Ki = 5.1 nM T16987 CLV5O9 122192682 Ki = 4.9 nM T16987 CH1N0C 122193189 Ki = 8050 nM T16987 C19HVL 122193190 Ki = 23100 nM T16987 C5TQJ1 122193251 Ki = 29200 nM T16987 C8XCL0 122193252 Ki = 10500 nM T16987 CH4IV8 122194771 Ki = 35.2 nM T16987 CQ7N0L 122194772 Ki = 44.9 nM T16987 CI5K2F 122194773 Ki = 8.3 nM T16987 CV51IU 122194774 Ki = 26.2 nM T16987 C7OFR6 122194775 Ki = 7.4 nM T16987 C81HNW 122194776 Ki = 81.1 nM T16987 C8J5QV 122194777 Ki = 77.2 nM T16987 CV1C9T 122194778 Ki = 7.3 nM T16987 CJC1W3 122194779 Ki = 6.7 nM T16987 CU1TV5 122194780 Ki = 237 nM T16987 C4C1BE 122194781 Ki = 93.9 nM T16987 CR9I5Q 122194782 Ki = 90.8 nM T16987 C8SVY4 122194783 Ki = 70.6 nM T16987 C7HT8B 122194784 Ki = 8.1 nM T16987 CW8P3R 122194785 Ki = 9.3 nM T16987 COAK34 122194786 Ki = 8.1 nM T16987 CPN73S 122199224 Ki = 4 nM T16987 C18KAD 122367673 Ki > 50000 nM T16987 CPN5F4 122367675 Ki > 50000 nM T16987 CGE1Q6 122707121 Ki = 0.58 nM T16987 C1JBF7 122707123 Ki = 760 nM T16987 CGPI62 123372490 Ki = 48.3 nM T16987 CV4GW7 126961712 Ki = 5.8 nM T16987 C0FD4E 126961713 Ki = 3.3 nM T16987 CXY79J 127024883 Ki = 4.9 nM T16987 CK9C7T 127024884 Ki = 4.3 nM T16987 C50MSQ 127024885 Ki = 5.6 nM T16987 C4N6WJ 127024886 Ki = 3.9 nM T16987 C5AES0 127024887 Ki = 4 nM T16987 CHU95V 127024991 Ki = 54.2 nM T16987 CP8O7D 127024992 Ki = 4.9 nM T16987 CRHW31 127024993 Ki = 65 nM T16987 C57BLH 127025130 Ki = 38.1 nM T16987 CRTB63 127025292 Ki = 19.5 nM T16987 CAO31Y 127025293 Ki = 38.3 nM T16987 CL0ZR4 127025295 Ki = 5.2 nM T16987 C9JNZ5 127025296 Ki = 96.7 nM T16987 C04USY 127025300 Ki = 0.6 nM T16987 CDB1Z9 127025301 Ki = 5.2 nM T16987 CYK6H1 127025302 Ki = 39.1 nM T16987 C7UF0B 127025480 Ki = 3.6 nM T16987 C6M4SW 127025591 Ki = 33.4 nM T16987 CUPA95 127025592 Ki = 1.5 nM T16987 CWP36V 127025593 Ki = 0.67 nM T16987 C95QVS 127026977 Ki = 8390 nM T16987 C09PAM 127026978 Ki = 5975 nM T16987 CS96JF 127026979 Ki = 9030 nM T16987 CRB80M 127026980 Ki = 7170 nM T16987 C0RBK5 127027010 Ki = 4.1 nM T16987 C0WY9H 127027097 Ki = 31.9 nM T16987 CP84DU 127027288 Ki = 6185 nM T16987 CH30BV 127027289 Ki = 75.1 nM T16987 CM72RV 127027290 Ki = 48.9 nM T16987 CO3IJ7 127027291 Ki = 15.5 nM T16987 C4O2XT 127028951 Ki = 4.5 nM T16987 CFIW54 127029020 Ki = 5.6 nM T16987 C5RBS3 127029021 Ki = 415 nM T16987 CPA6G5 127029022 Ki > 10000 nM T16987 C74ZGJ 127029023 Ki > 10000 nM T16987 CN3PH9 127029250 Ki = 5.5 nM T16987 CTY1H9 127029498 Ki = 17.8 nM T16987 C1J0RU 127029568 Ki = 0.6 nM T16987 CS2K4U 127034999 Ki = 0.74 nM T16987 CFG39M 127035855 Ki = 60.7 nM T16987 C6MH2V 127035856 Ki = 74.4 nM T16987 CVO4B6 127035857 Ki = 64.2 nM T16987 CQC6P9 127035858 Ki = 5.2 nM T16987 C7YA3N 127035859 Ki = 5 nM T16987 CXZI89 127035860 Ki = 0.66 nM T16987 C5KLP8 127035861 Ki = 6.8 nM T16987 CTVN28 127036466 Ki = 34.4 nM T16987 CWPY69 127036947 Ki = 68.6 nM T16987 CL76JS 127037630 Ki = 33.7 nM T16987 CY1JU3 127037755 Ki = 43.7 nM T16987 C0UQ7W 127037756 Ki = 57.4 nM T16987 CQUE67 127037757 Ki = 40.8 nM T16987 CL3Q0T 127037870 Ki = 55.6 nM T16987 CK3VW1 127037881 Ki = 33.9 nM T16987 CTSR32 127038212 Ki = 5.2 nM T16987 CQTS23 127038553 Ki = 32.2 nM T16987 CG8B3V 127039153 Ki = 44.4 nM T16987 CIO74C 127039154 Ki = 28.5 nM T16987 C0L8NH 127039155 Ki = 4.1 nM T16987 CS96GU 127039479 Ki = 48.9 nM T16987 C6WCG5 127039856 Ki = 2.2 nM T16987 C4NQ5H 127039905 Ki = 22.4 nM T16987 C3J8ET 127040041 Ki = 46.5 nM T16987 C0P5HB 127040227 Ki = 5.5 nM T16987 CCD87Q 127040239 Ki = 4.6 nM T16987 C97DAS 127040240 Ki = 5.5 nM T16987 C9OZP8 127040553 Ki = 35.3 nM T16987 C4SH5D 127040554 Ki = 2.7 nM T16987 CCO9S8 127040555 Ki = 32.6 nM T16987 C12SMV 127041490 Ki > 10000 nM T16987 CSJ3V0 127041732 Ki = 20.5 nM T16987 CG75VH 127041733 Ki = 10.7 nM T16987 CQC6A4 127042329 Ki = 56.4 nM T16987 CRZK01 127043469 Ki = 0.64 nM T16987 C41YOV 127044252 Ki = 0.9 nM T16987 CMTC13 127044428 Ki = 5.5 nM T16987 C7KU0Z 127044429 Ki = 3.7 nM T16987 CJO3U8 127044444 Ki = 1 nM T16987 CAXM67 127044445 Ki = 7.6 nM T16987 CHP23N 127044446 Ki = 7.2 nM T16987 C1T4LU 127044499 Ki = 7.11 nM T16987 CI3PD8 127044664 Ki = 0.61 nM T16987 CU5B2G 127044665 Ki = 0.73 nM T16987 CM9QJ3 127044834 Ki = 0.54 nM T16987 C5HIY4 127044835 Ki = 0.47 nM T16987 CKW0B5 127044836 Ki = 5.74 nM T16987 C4WZJ7 127044997 Ki = 0.66 nM T16987 C1LIQ5 127044998 Ki = 1.45 nM T16987 C3S2GY 127044999 Ki = 0.76 nM T16987 C1U0VA 127045339 Ki = 9.1 nM T16987 CG10PI 127048878 Ki = 2.5 nM T16987 C3PHY8 127048879 Ki = 14.31 nM T16987 COLX43 127048880 Ki = 55 nM T16987 CBJ74P 127048881 Ki = 13.26 nM T16987 C1XE4W 127049197 Ki = 3.42 nM T16987 CCX35L 127049198 Ki = 3.94 nM T16987 CRE6O9 127049213 Ki = 3.34 nM T16987 CP40EB 127049242 Ki = 3.7 nM T16987 CLFB54 127049248 Ki = 5.4 nM T16987 C5CNP8 127050174 Ki = 5.9 nM T16987 CH07TV 127050456 Ki = 0.54 nM T16987 CP8U0D 127050457 Ki = 0.54 nM T16987 C65PAS 127050458 Ki = 5.54 nM T16987 CJP49X 127050777 Ki = 0.61 nM T16987 CER02F 127050778 Ki = 3.16 nM T16987 CG17IO 127050812 Ki = 3.2 nM T16987 C8X6CY 127050822 Ki = 3.9 nM T16987 C4IA5N 127051119 Ki = 2.6 nM T16987 CRDQ30 127051120 Ki = 5.9 nM T16987 C5Y4DI 127051953 Ki = 2.8 nM T16987 CM21NF 127052276 Ki = 0.62 nM T16987 CI24ZM 127052900 Ki = 4.4 nM T16987 CEVZ36 127052901 Ki = 0.66 nM T16987 CX1Z2E 127052917 Ki = 4.23 nM T16987 CM8FI7 127052918 Ki = 24.56 nM T16987 CUOZ60 127052919 Ki = 38.42 nM T16987 C85FAK 129009671 Ki = 1.1 nM T16987 C7R6LY 129009672 Ki = 1.1 nM T16987 C2B6XM 129673327 Ki = 7.6 nM T16987 CJC35Q 129856021 Ki = 34.7 nM T16987 CCF61S 129883275 Ki = 40.8 nM T16987 C7Z4UB 132494202 Ki = 818.7 nM T16987 C20FGA 132495363 Ki = 6.7 nM T16987 C4GR3Y 132498655 Ki = 8.6 nM T16987 CVM1A9 132547283 Ki = 3.3 nM T16987 C3H1NS 132547284 Ki = 3.8 nM T16987 C1FWS2 132547285 Ki = 75.6 nM T16987 C7Z5LX 132547286 Ki = 62.1 nM T16987 CW97YT 132547287 Ki = 4.1 nM T16987 CW18RT 132547288 Ki = 147 nM T16987 COC54I 132547289 Ki = 297 nM T16987 CX4DM9 132547290 Ki = 23.8 nM T16987 C5JM7W 132547291 Ki = 22.3 nM T16987 C7V6XS 132547292 Ki = 362 nM T16987 CRL24F 132596304 Ki = 670 nM T16987 C6OA8Z 132819872 Ki = 0.82 nM T16987 CJGH58 132819873 Ki = 8.4 nM T16987 COT92G 132819874 Ki = 1.5 nM T16987 COS36W 132819875 Ki = 5.2 nM T16987 CMAU69 132819876 Ki = 17.1 nM T16987 CY62CQ 132938107 Ki = 0.57 nM T16987 CB8T7K 132938108 Ki = 1.9 nM T16987 CY6L7Z 132941396 Ki = 6.8 nM T16987 CEP32W 132991412 Ki = 10.2 nM T16987 CG0HL2 134130044 Ki = 79.4 nM T16987 C63CQL 134130121 Ki = 26.7 nM T16987 C82HUT 134130285 Ki = 84.8 nM T16987 CMZ76O 134130322 Ki = 302 nM T16987 C8AL2D 134130377 Ki = 80.1 nM T16987 C7N0JD 134130389 Ki = 359 nM T16987 CZ7CA3 134131127 Ki = 50.4 nM T16987 C5XU9Y 134131319 Ki = 35.1 nM T16987 CZ2YK7 134131524 Ki = 41.4 nM T16987 CUVB06 134131580 Ki = 48.1 nM T16987 C94HZF 134131659 Ki = 1.1 nM T16987 CU5B8H 134131865 Ki = 1.1 nM T16987 C2UIM6 134132835 Ki = 7.8 nM T16987 CECZ43 134133137 Ki = 10.5 nM T16987 C83QKJ 134133977 Ki = 7.1 nM T16987 CJ3EQ2 134136523 Ki = 3.2 nM T16987 C4IO1K 134137058 Ki = 12.9 nM T16987 CWG0L5 134139228 Ki = 101.6 nM T16987 CJ4R6E 134141819 Ki = 8.8 nM T16987 CBK73M 134146037 Ki = 1 nM T16987 CDH38B 134147400 Ki = 4.3 nM T16987 CDSM29 134147656 Ki = 80.1 nM T16987 C1Q8GK 134149666 Ki = 4.9 nM T16987 CF31OS 134149711 Ki = 12.9 nM T16987 C2NXB7 134151324 Ki = 8.2 nM T16987 CR4VE0 134152281 Ki = 8.9 nM T16987 CU0T4X 134152542 Ki = 5.4 nM T16987 CZ9C1N 134152694 Ki = 5.9 nM T16987 C4WBC6 134153047 Ki = 6 nM T16987 CSK6L9 134154625 Ki = 10.2 nM T16987 CG69UV 134155483 Ki = 12.1 nM T16987 C19BHQ 134817796 Ki = 5.7 nM T16987 CY3E4D 134817797 Ki = 48 nM T16987 C8IF6V 134817798 Ki = 7.3 nM T16987 C0UL7A 134828600 Ki = 950 nM T16987 C4ZLP6 134828601 Ki = 80 nM T16987 C3OLP6 134828602 Ki = 880 nM T16987 CJT9W0 135393499 Ki = 6.6 nM T16987 CK8FP3 135393500 Ki = 7.8 nM T16987 CRL4V7 135393501 Ki = 5.6 nM T16987 CTR37Z 135408753 Ki = 10460 nM T16987 C4CXD1 135434964 Ki = 30.1 nM T16987 CFK9A4 135434965 Ki = 11.9 nM T16987 CY7RT4 135442220 Ki = 320 nM T16987 CKAF26 135460193 Ki = 24 nM T16987 C0WEU9 135537166 Ki = 2.8 nM T16987 CC8IO3 135595465 Ki = 1950 nM T16987 C74TBX 135595467 Ki = 2142 nM T16987 CX1NF7 135595474 Ki = 397 nM T16987 CL71ND 135645043 Ki = 41000 nM T16987 C1WH3Z 135891810 Ki = 8.3 nM T16987 CSH8M1 135995959 Ki = 7.4 nM T16987 CB90PQ 135995960 Ki = 6.7 nM T16987 CNG0L4 136044222 Ki = 58.5 nM T16987 CQ02AW 136044223 Ki = 498 nM T16987 C47KQP 136053622 Ki = 11.6 nM T16987 C1M7DN 136053656 Ki = 1.62 nM T16987 C4A2XS 136198631 Ki = 9.91 nM T16987 C93PWB 136198632 Ki = 85.83 nM T16987 CVME35 136198643 Ki = 1107 nM T16987 CBO5I1 136242872 Ki = 9.2 nM T16987 CQDT25 136242873 Ki = 7.8 nM T16987 CK5AZ7 136242878 Ki = 9.1 nM T16987 C1NTA3 136418497 Ki = 58.6 nM T16987 C6VS7N 136607460 Ki = 0.9 nM T16987 CAC75Q 136607461 Ki = 0.83 nM T16987 CI28TM 136934908 Ki = 837 nM T16987 C9UKC8 136998786 Ki = 438 nM T16987 C3QFS1 136998787 Ki = 143 nM T16987 C1P9FJ 136998788 Ki = 55.5 nM T16987 CZ40LF 137028501 Ki = 91.5 nM T16987 C5Q8PD 137028502 Ki = 65.9 nM T16987 CSL47A 137028503 Ki = 83.6 nM T16987 C7T1HR 137028504 Ki = 244 nM T16987 C9WH2P 137028505 Ki = 73.5 nM T16987 CGBQ10 137028506 Ki = 44.5 nM T16987 C4DHG6 137028507 Ki = 91.4 nM T16987 CIP84X 137028508 Ki = 74.6 nM T16987 CF14KA 137028511 Ki = 3.7 nM T16987 CXHB30 137028512 Ki = 6.5 nM T16987 CRMC05 137028513 Ki = 37.7 nM T16987 CJH4E5 137028514 Ki = 22.8 nM T16987 CGAR93 137028515 Ki = 56.8 nM T16987 C4QG2K 137028516 Ki = 82.8 nM T16987 C2GMH5 137028517 Ki = 5.4 nM T16987 CBX6S7 137028518 Ki = 7.2 nM T16987 CUW85H 137062187 Ki = 0.67 nM T16987 C4XY9S 137091066 Ki = 2.32 nM T16987 C64ITR 137091070 Ki = 2.83 nM T16987 C0BEH8 137093138 Ki = 624 nM T16987 CD6C0A 137093141 Ki = 14600 nM T16987 CE9QV3 137226330 Ki = 66.7 nM T16987 C4SMA5 137226331 Ki = 62.5 nM T16987 C2H6VC 137226372 Ki = 2.31 nM T16987 CZY9D7 137226374 Ki = 1.76 nM T16987 C6YBD3 137226375 Ki = 0.69 nM T16987 C7DMR8 137226384 Ki = 0.64 nM T16987 C2KG3D 137226385 Ki = 1.17 nM T16987 C0KMB4 137226399 Ki = 0.54 nM T16987 CD1VC9 137226400 Ki = 0.58 nM T16987 C4F8NU 137226401 Ki = 0.69 nM T16987 CW65FQ 137226402 Ki = 0.63 nM T16987 CY95JF 137226420 Ki = 0.47 nM T16987 CW52IQ 137631447 Ki = 8700 nM T16987 CZ5GQ4 137631746 Ki = 80.7 nM T16987 CFQ5W2 137631798 Ki > 50000 nM T16987 C7O3CP 137632017 Ki = 10100 nM T16987 CN8UL1 137632214 Ki = 10100 nM T16987 CH42MU 137632574 Ki = 727.5 nM T16987 CL5K3D 137632743 Ki = 92.6 nM T16987 CE20FG 137632898 Ki > 50000 nM T16987 CO25DP 137632949 Ki = 9.1 nM T16987 CFE79H 137633320 Ki = 86.4 nM T16987 C9AD2H 137633797 Ki > 50000 nM T16987 CVNO32 137633860 Ki = 84.6 nM T16987 C0P6ZT 137634762 Ki = 46.9 nM T16987 CS6M2N 137635469 Ki = 546 nM T16987 CNJV53 137635486 Ki = 4700 nM T16987 CZ4Q1T 137636083 Ki = 10.5 nM T16987 C9GIX7 137636130 Ki > 50000 nM T16987 CV12YX 137636350 Ki > 100 nM T16987 CE46DY 137636432 Ki = 45.2 nM T16987 CK0N2Y 137636453 Ki = 59 nM T16987 CM9YC2 137636494 Ki = 10.6 nM T16987 CMX9T3 137636945 Ki = 10900 nM T16987 C7YKB0 137636981 Ki > 50000 nM T16987 C2Z7GO 137637071 Ki = 847 nM T16987 CWO5Z6 137637365 Ki > 100 nM T16987 CQ5K1H 137637688 Ki = 6 nM T16987 C2HY8G 137637767 Ki > 50000 nM T16987 CK6OW4 137638637 Ki = 13 nM T16987 C6V8ED 137638882 Ki = 19.7 nM T16987 C64JQN 137639095 Ki = 4.3 nM T16987 CVJ35I 137639180 Ki = 8300 nM T16987 C12QYH 137639189 Ki = 1000 nM T16987 C29XAH 137639434 Ki = 84.4 nM T16987 CH2C3F 137639611 Ki = 4.9 nM T16987 CPR04H 137639655 Ki = 4.7 nM T16987 C4SP7Q 137639785 Ki = 80.5 nM T16987 C2OT9R 137640310 Ki > 50000 nM T16987 C5OU2V 137640459 Ki = 19.9 nM T16987 C8P3SC 137640892 Ki = 722.7 nM T16987 CJ4M2A 137640917 Ki = 47.2 nM T16987 CR65OQ 137640944 Ki = 43.1 nM T16987 C75WMG 137641075 Ki = 9570 nM T16987 C6B0CQ 137641198 Ki = 4.3 nM T16987 C0HER8 137641290 Ki > 50000 nM T16987 CR2MU6 137641422 Ki > 50000 nM T16987 CMOZ57 137641425 Ki > 50000 nM T16987 CCSN50 137642054 Ki = 6.5 nM T16987 CN6WS9 137642180 Ki > 50000 nM T16987 C0Z9DH 137642233 Ki > 50000 nM T16987 C7ZX8Q 137643203 Ki > 50000 nM T16987 C3Y2GU 137643607 Ki > 50000 nM T16987 C0B8QA 137643949 Ki > 100 nM T16987 CG13TO 137643998 Ki = 5900 nM T16987 CIK49D 137644678 Ki = 4.2 nM T16987 CV75NJ 137644865 Ki = 723.6 nM T16987 CWQ91B 137644949 Ki = 12 nM T16987 CV0AH9 137645517 Ki = 26 nM T16987 CFV6T3 137645790 Ki > 50000 nM T16987 C3CI0M 137645793 Ki = 8 nM T16987 C7E6NL 137646223 Ki > 50000 nM T16987 C10YVU 137646329 Ki > 50000 nM T16987 CRP78K 137647221 Ki > 100 nM T16987 CXD9A0 137647636 Ki = 7.6 nM T16987 CR2H7M 137647845 Ki > 50000 nM T16987 CY15KD 137648125 Ki = 61.3 nM T16987 C5PEA6 137648128 Ki = 23.4 nM T16987 CU81DA 137648494 Ki = 7.6 nM T16987 C82NJP 137648964 Ki = 10800 nM T16987 CGLM50 137649870 Ki = 5.8 nM T16987 C2HA7Q 137649882 Ki = 892 nM T16987 C4N1MP 137650156 Ki = 6.7 nM T16987 CCZ4N1 137650188 Ki = 9300 nM T16987 C1FO3T 137650198 Ki = 2.4 nM T16987 C91KQA 137650256 Ki = 2.6 nM T16987 C5V6XP 137651635 Ki = 3.2 nM T16987 CSTP12 137651755 Ki = 3 nM T16987 C01BXO 137651769 Ki = 59.1 nM T16987 CY0C6Z 137652226 Ki = 57.8 nM T16987 C6GWB1 137652305 Ki = 7.7 nM T16987 C5DG1K 137652445 Ki = 1.7 nM T16987 CN0W6U 137653170 Ki > 50000 nM T16987 C9UGN4 137653309 Ki > 50000 nM T16987 C45WNI 137653361 Ki > 50000 nM T16987 C4U9KA 137653686 Ki = 1000 nM T16987 CNJ6P9 137654601 Ki = 6.1 nM T16987 CRC23M 137655132 Ki = 31.6 nM T16987 CWT49Q 137655252 Ki = 13600 nM T16987 C2P5FH 137655445 Ki > 50000 nM T16987 C3DT7S 137655450 Ki > 100 nM T16987 CASB61 137655528 Ki = 5.9 nM T16987 C0XPN2 137655580 Ki = 39.9 nM T16987 CUO84H 137655694 Ki = 732.4 nM T16987 CHD58S 137656247 Ki = 74.6 nM T16987 CRXD65 137656549 Ki = 6600 nM T16987 CG5EK0 137656938 Ki = 445 nM T16987 CT7CW2 137657041 Ki = 10900 nM T16987 C3PAQ7 137657121 Ki = 920 nM T16987 C2SYC9 137657578 Ki = 60 nM T16987 C8RNZ6 137657759 Ki = 39 nM T16987 CTI2V7 137658103 Ki = 961 nM T16987 CH39CL 137658251 Ki = 3.5 nM T16987 CL2H0T 137658375 Ki = 80.8 nM T16987 C7V6MY 137658589 Ki = 9.8 nM T16987 CT98MV 137658877 Ki > 100 nM T16987 C8YV5D 137659052 Ki = 9.3 nM T16987 CXO9Y7 137659205 Ki = 81.7 nM T16987 CJ5O8M 137659269 Ki > 50000 nM T16987 C40MRZ 137659514 Ki > 50000 nM T16987 CCX48V 137659570 Ki = 36.7 nM T16987 CXK83H 137659797 Ki = 74.1 nM T16987 CHKB25 137659801 Ki > 10000 nM T16987 CQ56MJ 137661167 Ki = 9.7 nM T16987 CF6Z9A 137661353 Ki = 23.9 nM T16987 CRC92Y 137661359 Ki = 933 nM T16987 CN1JH4 137661469 Ki = 4.9 nM T16987 C1Z8KG 137661675 Ki = 4.7 nM T16987 CEAR56 137662187 Ki > 50000 nM T16987 CO8UE3 137662293 Ki = 47.7 nM T16987 C08ZTR 138393077 Ki = 7.6 nM T16987 CIX41M 138393379 Ki = 53.7 nM T16987 CBOM51 138753317 Ki = 42.8 nM T16987 C8TWF0 139597735 Ki = 80 nM T16987 CR10ZH 139823666 Ki > 1000 nM T16987 C78UAW 142468585 Ki = 174 nM T16987 CZY8Q6 142468589 Ki = 0.56 nM T16987 C3HMI0 142468591 Ki = 219 nM T16987 CHA65U 142468595 Ki > 50000 nM T16987 C6KE9A 142468600 Ki > 50000 nM T16987 C65DHJ 142468602 Ki = 43.2 nM T16987 CI02LX 142468604 Ki > 50000 nM T16987 C7LP3J 142468605 Ki > 50000 nM T16987 CA9O2I 142468608 Ki = 471 nM T16987 CUE58A 142547533 Ki = 7.8 nM T16987 C6GB9T 143032987 Ki = 0.97 nM T16987 CNW7H1 145948231 Ki = 6.5 nM T16987 C3PF4Q 145948234 Ki = 7.3 nM T16987 CI9H2E 145949226 Ki = 583.2 nM T16987 CP6AM5 145949377 Ki = 18.1 nM T16987 CGLD54 145949403 Ki = 8.9 nM T16987 CROP78 145949554 Ki = 23.8 nM T16987 CSW7B8 145950055 Ki = 706.1 nM T16987 C7DBT4 145950298 Ki = 87.4 nM T16987 CJSK40 145950390 Ki = 342.9 nM T16987 C2H9QY 145950512 Ki = 183.3 nM T16987 C7BK9O 145950527 Ki = 87.5 nM T16987 C63SMQ 145950568 Ki = 31 nM T16987 CE58JF 145950709 Ki = 49.9 nM T16987 C8XAH1 145950880 Ki = 4.1 nM T16987 C53EGH 145950894 Ki = 1.6 nM T16987 C8IGY9 145950981 Ki = 5.5 nM T16987 C87JIM 145951255 Ki = 44.4 nM T16987 CL25SI 145951508 Ki = 646.5 nM T16987 CJ2W6V 145951720 Ki = 2.8 nM T16987 CQC79A 145951865 Ki = 164.1 nM T16987 CKZT53 145951931 Ki = 4529.4 nM T16987 C3R8NQ 145951979 Ki = 337.9 nM T16987 CGFU20 145952201 Ki = 359.8 nM T16987 CUJ2G6 145952345 Ki = 1.5 nM T16987 CU69PG 145952370 Ki = 64.6 nM T16987 CWE6M8 145952775 Ki = 731.9 nM T16987 CUB49H 145952983 Ki = 24.7 nM T16987 CNZX07 145953044 Ki = 44.9 nM T16987 C1KQ3D 145953178 Ki = 225.8 nM T16987 C7Q4IN 145953662 Ki = 357.1 nM T16987 C7GIQ5 145954093 Ki = 6400 nM T16987 CM4U3B 145954289 Ki = 31.1 nM T16987 C67HYG 145954632 Ki > 10000 nM T16987 CTV8L5 145954775 Ki > 10000 nM T16987 C0UBV8 145955012 Ki = 27.7 nM T16987 C7QL4I 145955037 Ki = 78.8 nM T16987 CM9Y2S 145955268 Ki = 3.4 nM T16987 CI64UX 145955888 Ki = 9 nM T16987 C9DLX6 145955997 Ki = 737.2 nM T16987 CMGN62 145956070 Ki = 82.2 nM T16987 CS93JU 145956073 Ki = 72.4 nM T16987 CHXP91 145956144 Ki = 2.4 nM T16987 CZK0L8 145956164 Ki = 1.9 nM T16987 CQJO72 145956348 Ki = 33.3 nM T16987 CAPD95 145956503 Ki = 7.7 nM T16987 CRYP47 145956664 Ki = 818.7 nM T16987 CE39IU 145956732 Ki = 89.1 nM T16987 CYH7O8 145956770 Ki = 369.2 nM T16987 CRUI17 145956819 Ki = 58.6 nM T16987 C6I1XE 145956976 Ki = 41.9 nM T16987 C7X6NA 145957099 Ki = 91.9 nM T16987 CKOX92 145957394 Ki = 392.8 nM T16987 C98PXC 145957555 Ki = 73.4 nM T16987 CI5B9M 145957665 Ki = 27.3 nM T16987 C6JL8X 145958066 Ki = 77.6 nM T16987 CQO8H5 145958250 Ki = 2.8 nM T16987 CC32ZJ 145958632 Ki = 4.9 nM T16987 C14UQR 145958824 Ki = 9.3 nM T16987 C2MCO8 145958917 Ki = 7.8 nM T16987 C37CVT 145959395 Ki = 737.2 nM T16987 CM5OK6 145959413 Ki = 255.5 nM T16987 C7J6MA 145959539 Ki = 359.8 nM T16987 CK8DX1 145959911 Ki = 6062.5 nM T16987 C29YFS 145959974 Ki = 39.8 nM T16987 C9MSK2 145960116 Ki = 1.5 nM T16987 CB49ZJ 145960257 Ki = 671.9 nM T16987 C3JTG4 145960436 Ki = 6.2 nM T16987 CVMF36 145960835 Ki = 6.8 nM T16987 CBGV25 145960853 Ki = 34 nM T16987 CD2X3F 145961133 Ki = 7.5 nM T16987 CBT85V 145961452 Ki = 6.8 nM T16987 CCYK28 145962259 Ki = 5.2 nM T16987 CQV18P 145962416 Ki = 11.6 nM T16987 C34BRN 145962803 Ki = 28.4 nM T16987 C36LCF 145962935 Ki = 3.6 nM T16987 CZ9PL4 145963030 Ki = 47.7 nM T16987 CGY68S 145963294 Ki = 6.3 nM T16987 CJU15K 145963586 Ki = 6.7 nM T16987 CVL39I 145963679 Ki = 53.8 nM T16987 CUZ3A5 145963719 Ki = 5 nM T16987 CM71JT 145964104 Ki = 7.4 nM T16987 CGTA80 145964130 Ki = 94.1 nM T16987 C4C9IE 145964340 Ki = 7 nM T16987 CK21BE 145964400 Ki = 57.6 nM T16987 CAPU84 145964558 Ki = 4.1 nM T16987 CGR16W 145965551 Ki = 210 nM T16987 CWHV36 145965762 Ki = 310 nM T16987 CCDI76 145966475 Ki = 6.5 nM T16987 CMF72D 145966553 Ki = 7.6 nM T16987 CQ64RX 145966558 Ki = 35 nM T16987 CJ4D0R 145967030 Ki = 68.6 nM T16987 C7SUX3 145967040 Ki = 59.2 nM T16987 CDYR51 145968242 Ki = 93.8 nM T16987 CKME70 145968701 Ki = 7.5 nM T16987 CX4D2R 145969379 Ki = 7.3 nM T16987 C6DQK4 145972104 Ki = 4.2 nM T16987 CYMF38 145972316 Ki = 43.3 nM T16987 CD42QZ 145972397 Ki = 2.9 nM T16987 CF5KR4 145972986 Ki = 64 nM T16987 C9MZS1 145973465 Ki = 65 nM T16987 C8UAD6 145973595 Ki = 2.4 nM T16987 CX5U8J 145974401 Ki = 5.2 nM T16987 CJD0I1 145974412 Ki = 340 nM T16987 C1QZ7F 145974710 Ki = 94.4 nM T16987 CDU4M5 145975077 Ki = 8.6 nM T16987 C3I2WU 145975151 Ki = 90.2 nM T16987 CBL8Y4 145975424 Ki = 5 nM T16987 CPK17Y 145975721 Ki = 350 nM T16987 CZVK21 145975933 Ki = 93.5 nM T16987 CO9M3B 145976300 Ki = 280 nM T16987 CI9C6U 145976539 Ki = 92.8 nM T16987 CHI26Q 145976735 Ki = 90.3 nM T16987 CZWC63 145977536 Ki = 44 nM T16987 CUEB47 145977814 Ki = 27.2 nM T16987 CK9L7E 145977947 Ki = 25.8 nM T16987 C69UQY 145978025 Ki = 84.1 nM T16987 CO0J6L 145978583 Ki = 86.4 nM T16987 CYG69V 145978605 Ki = 54 nM T16987 CYWK54 145978673 Ki = 6.6 nM T16987 CA32BT 145978780 Ki = 19.4 nM T16987 CXI41R 145978938 Ki = 160 nM T16987 CM8KP7 145979094 Ki = 500 nM T16987 C82LKO 145979169 Ki = 90 nM T16987 CI34JB 145979332 Ki = 43.3 nM T16987 COYX31 145979594 Ki = 9.6 nM T16987 CXDE63 145979618 Ki = 780 nM T16987 C7ZOM8 145979619 Ki = 60 nM T16987 CMT6G7 145979772 Ki = 78.1 nM T16987 C9H6AW 145979979 Ki = 340 nM T16987 CS85AP 145980216 Ki = 840 nM T16987 CWA24U 145980366 Ki = 40.2 nM T16987 C85TGI 145980938 Ki = 9.6 nM T16987 C97LPB 145981035 Ki = 15.3 nM T16987 C1RO4L 145981799 Ki = 210 nM T16987 C4DNF7 145982126 Ki = 16.7 nM T16987 C7N6RT 145982437 Ki = 8.7 nM T16987 C3J5NQ 145983899 Ki = 24.7 nM T16987 CTZ71U 145986436 Ki = 460 nM T16987 CIDO62 145986509 Ki = 620 nM T16987 CK05FT 145986641 Ki = 310 nM T16987 CG6CU5 145987209 Ki = 6.9 nM T16987 CT01AM 145987366 Ki = 220 nM T16987 CI9F3V 145987533 Ki = 24.7 nM T16987 CQF4O8 145987804 Ki = 53.1 nM T16987 CBF3V2 145987828 Ki = 57.8 nM T16987 C0LVN9 145987839 Ki = 53.9 nM T16987 C8XDH5 145988129 Ki = 530 nM T16987 CO3N6M 145988784 Ki = 5.2 nM T16987 CPZN93 145988792 Ki = 44.1 nM T16987 CZW72V 145988876 Ki = 5.5 nM T16987 C39ZMI 145988963 Ki = 3 nM T16987 C7AUF1 145989028 Ki = 69 nM T16987 C6BKP8 145989063 Ki = 70 nM T16987 C35VEG 145989087 Ki = 800 nM T16987 C6DN9E 145989219 Ki = 650 nM T16987 COZM89 145989422 Ki = 300 nM T16987 CJH51I 145989433 Ki = 300 nM T16987 CA8K2J 145990039 Ki = 65.6 nM T16987 C8XD2V 145990044 Ki = 830 nM T16987 CLQ12A 145990129 Ki = 35.9 nM T16987 CJQ73W 145990589 Ki = 48.7 nM T16987 C2WTN6 145990640 Ki = 70.4 nM T16987 CM6SA4 145990881 Ki = 44.1 nM T16987 CIA37P 145991377 Ki = 7.1 nM T16987 CWH89P 145991839 Ki = 8 nM T16987 C58FGU 145992776 Ki = 250 nM T16987 CH48GI 145992962 Ki = 6.6 nM T16987 CO42RK 145992983 Ki = 9 nM T16987 C8IE2X 145993014 Ki = 9.1 nM T16987 CDC84X 145993019 Ki = 5.8 nM T16987 CE0HY6 145993300 Ki = 43.5 nM T16987 CMS86X 145993352 Ki = 790 nM T16987 CB12JK 145993432 Ki = 44.7 nM T16987 CZSC36 145993499 Ki = 9.2 nM T16987 CEC07M 145993642 Ki = 530 nM T16987 CIDP76 145994238 Ki = 7.8 nM T16987 C48CZD 146160385 Ki = 30.8 nM T16987 C2SG4L 146833326 Ki = 86.8 nM T16987 C6FD2N 147348395 Ki = 34.6 nM T16987 CGMX98 155510724 Ki = 0.9 nM T16987 C3QJI5 155510851 Ki = 9.3 nM T16987 CY5T1K 155510897 Ki = 659.3 nM T16987 CN6DW9 155511075 Ki = 35.7 nM T16987 C2PXC3 155511133 Ki = 0.8 nM T16987 C1A5OB 155511232 Ki = 88.3 nM T16987 C30ADE 155511364 Ki = 2725 nM T16987 C1D8JF 155511459 Ki > 10000 nM T16987 C6QNX5 155511723 Ki = 3.3 nM T16987 C03BJU 155511800 Ki = 750 nM T16987 CMCL94 155512138 Ki = 67.6 nM T16987 CI40CL 155512225 Ki = 25.3 nM T16987 C7J0HP 155512942 Ki > 100000 nM T16987 C51PHM 155512962 Ki = 60.6 nM T16987 CN53ED 155512974 Ki > 100000 nM T16987 CVSG61 155513076 Ki = 105.1 nM T16987 CW1DP7 155513481 Ki = 27.3 nM T16987 C7QT4V 155513609 Ki = 7.6 nM T16987 CX2UJ9 155514131 Ki = 3900 nM T16987 CV7WR4 155514243 Ki = 8.9 nM T16987 C67VGD 155514389 Ki = 9.4 nM T16987 C7W9NI 155514825 Ki = 466 nM T16987 CU9H2A 155514935 Ki = 31 nM T16987 CMQV46 155514970 Ki = 22.3 nM T16987 CR89MP 155515069 Ki = 24.1 nM T16987 CW08ZX 155515305 Ki = 650 nM T16987 C5IPM8 155515308 Ki = 8 nM T16987 C46UNX 155515514 Ki = 9.2 nM T16987 C6DG3E 155515525 Ki > 100000 nM T16987 C7MER6 155515557 Ki = 710 nM T16987 C7UQ3J 155515746 Ki = 733 nM T16987 CT2ZB0 155515980 Ki = 8.5 nM T16987 C74SEH 155516204 Ki > 100000 nM T16987 CM9F7H 155516281 Ki > 50000 nM T16987 CLNT85 155516404 Ki = 3.8 nM T16987 COP4Q6 155516517 Ki = 728.1 nM T16987 C9LWV6 155516550 Ki = 21.6 nM T16987 C7IR3P 155516553 Ki = 5700 nM T16987 CBV6D3 155516701 Ki = 51.4 nM T16987 CP0NH3 155516885 Ki > 10000 nM T16987 CAG9L4 155517430 Ki = 9.6 nM T16987 C3OW4N 155517544 Ki > 50000 nM T16987 CW18JG 155517622 Ki = 827.8 nM T16987 C2H3JR 155517687 Ki > 100000 nM T16987 CQI20B 155517798 Ki > 100000 nM T16987 CRP2A6 155517861 Ki = 55.9 nM T16987 CWP3G6 155517862 Ki > 10000 nM T16987 CF07ZS 155517996 Ki = 31 nM T16987 C0O5CN 155518098 Ki > 10000 nM T16987 CUN49T 155518138 Ki = 16.2 nM T16987 C92QDE 155518180 Ki = 34.2 nM T16987 C1VNX3 155518220 Ki = 24.6 nM T16987 CP0U8D 155518225 Ki > 50000 nM T16987 CP7UI1 155518510 Ki = 42 nM T16987 CHI59Y 155518875 Ki = 7500 nM T16987 CL92UI 155519026 Ki = 20.8 nM T16987 C5TO4Q 155519047 Ki > 100000 nM T16987 CRF95N 155519064 Ki = 940.3 nM T16987 CI84OL 155519083 IC50 = 270 nM T16987 CN8RC2 155519138 Ki = 570 nM T16987 CK21TJ 155519240 Ki = 20.5 nM T16987 C8MYG2 155519248 Ki = 26.7 nM T16987 CO6D1Y 155519288 Ki = 34.1 nM T16987 CT56OD 155519473 Ki = 8.7 nM T16987 CI18TP 155519626 Ki = 569.6 nM T16987 CP4IL9 155519983 Ki = 29.6 nM T16987 CIV68R 155520019 Ki = 22.4 nM T16987 C5PN0D 155520029 Ki = 66.5 nM T16987 C1AQP3 155520260 IC50 = 3700 nM T16987 CP49HE 155520274 Ki = 8.6 nM T16987 C4Z8MX 155520314 Ki = 39 nM T16987 C5JCL6 155520507 Ki = 44.5 nM T16987 CG4VJ8 155520652 Ki = 680 nM T16987 C80OQU 155520908 Ki > 50000 nM T16987 C9Z1FL 155521038 Ki = 66.4 nM T16987 C2J1YG 155521041 Ki = 19.7 nM T16987 C2PR8W 155521294 Ki = 32.9 nM T16987 CN2X1Q 155521353 Ki = 10.2 nM T16987 CB54YX 155521489 Ki = 10.1 nM T16987 CRQ4L3 155521766 Ki = 85.2 nM T16987 CNP87G 155521876 Ki = 69.2 nM T16987 CR49AJ 155521885 Ki = 8.8 nM T16987 C4IYX7 155521930 Ki = 97.6 nM T16987 C2Q7BG 155522085 Ki = 61.3 nM T16987 C0A4EO 155522100 Ki = 21.9 nM T16987 CSN4C2 155522321 Ki = 462.6 nM T16987 C70NUX 155522372 Ki = 80.9 nM T16987 C8K9OI 155522618 Ki = 10.1 nM T16987 CDN9Z5 155522816 Ki = 63.7 nM T16987 C0Z3QT 155522883 Ki = 61.1 nM T16987 CJ49ZN 155522995 Ki = 42 nM T16987 CA9F2I 155523252 Ki = 98.5 nM T16987 C2XUA7 155523274 IC50 = 170 nM T16987 C3HGK6 155523328 Ki = 20.9 nM T16987 C6YZM3 155523403 Ki > 100 nM T16987 C9Q2WR 155523406 Ki = 219.3 nM T16987 CU2N9J 155523547 Ki = 11.8 nM T16987 CIF91M 155523572 Ki = 7.8 nM T16987 C9LF7B 155523634 Ki > 100000 nM T16987 C4U8XN 155523810 Ki = 33.8 nM T16987 CWD9Y1 155523853 Ki = 10.1 nM T16987 C0MZ5G 155524206 Ki = 8.5 nM T16987 C6KCG7 155524248 Ki > 50000 nM T16987 CK86ZT 155524367 Ki = 0.88 nM T16987 CK80AQ 155524610 Ki = 74.4 nM T16987 CDO4X2 155524724 Ki = 105 nM T16987 C3DM5L 155524759 Ki = 932.7 nM T16987 C5J8AS 155524785 Ki = 33.7 nM T16987 CS0WP1 155524852 Ki = 16400 nM T16987 C8M1KI 155525036 Ki = 47.1 nM T16987 CV6N0C 155525231 Ki = 19.9 nM T16987 CHT29F 155525313 Ki = 827.1 nM T16987 C4R1OT 155526288 Ki = 89.8 nM T16987 CGC8Y0 155526420 Ki = 9.2 nM T16987 CKT14B 155526554 Ki = 42.3 nM T16987 C0XZD3 155526695 Ki > 50000 nM T16987 CWGS97 155526825 Ki = 52.6 nM T16987 CGV91K 155527018 Ki = 73.6 nM T16987 CCL7V8 155527060 Ki = 415.3 nM T16987 CNVX86 155527078 Ki = 103.9 nM T16987 CG8JZ9 155527153 Ki = 10.2 nM T16987 C8K3OI 155527167 Ki = 6.3 nM T16987 C1LDV0 155527209 Ki = 49.7 nM T16987 C1I5PO 155527240 Ki > 50000 nM T16987 CK8XN6 155527284 Ki = 60.9 nM T16987 C4N7OY 155527400 Ki = 32.1 nM T16987 CJ3K9W 155527428 Ki = 38.9 nM T16987 C7YW9E 155527622 Ki > 50000 nM T16987 C65FOA 155527703 Ki = 16.5 nM T16987 C07LVI 155527781 Ki = 50.2 nM T16987 CPAH30 155527788 Ki = 16.3 nM T16987 C5XC7V 155527967 Ki = 2899 nM T16987 CDN05K 155527975 Ki = 87.3 nM T16987 C0RJ2M 155528294 Ki = 17.6 nM T16987 CN9G0E 155528332 Ki = 910 nM T16987 C4IML7 155528345 Ki = 76.9 nM T16987 C5X0CS 155528825 Ki > 100000 nM T16987 C7DCG0 155529026 Ki = 15.7 nM T16987 C1T2EA 155529101 Ki = 34.4 nM T16987 CWEQ38 155529122 Ki = 36.7 nM T16987 C52QUD 155529352 Ki = 0.86 nM T16987 CG94RZ 155529376 Ki = 803.6 nM T16987 C6TQ7W 155529566 IC50 = 2330 nM T16987 C2NY1E 155529877 Ki = 23 nM T16987 C2JV7R 155529885 Ki = 404 nM T16987 CJ21OD 155530289 Ki > 50000 nM T16987 CKO2V5 155530358 Ki = 49.2 nM T16987 C7TV5H 155530408 Ki = 45.2 nM T16987 C9Y4VC 155530502 Ki = 9.7 nM T16987 CTJ3I7 155530506 Ki = 49.4 nM T16987 C0HQ8E 155530537 Ki = 8.9 nM T16987 CP3UJ0 155530687 Ki = 9.5 nM T16987 C2T0LQ 155530848 Ki = 1.9 nM T16987 C3GK9H 155530900 Ki = 30.8 nM T16987 C2MT3K 155530925 Ki = 56.4 nM T16987 C8C4BT 155531090 Ki > 50000 nM T16987 CICU68 155531183 Ki = 0.76 nM T16987 CGN43T 155531186 Ki = 7.2 nM T16987 CO7P5W 155531268 Ki = 6.4 nM T16987 CLMZ93 155531382 Ki = 58.1 nM T16987 CYBD02 155531537 Ki = 1623 nM T16987 C43LZI 155531630 Ki = 6.9 nM T16987 CC5L6V 155531813 Ki = 9.2 nM T16987 CFV23M 155531820 Ki > 100000 nM T16987 CUM2B8 155532026 Ki = 8800 nM T16987 C83DJY 155532441 Ki > 100000 nM T16987 CASV53 155532466 Ki = 9.6 nM T16987 CFK8R5 155532512 Ki > 100000 nM T16987 CH6QB8 155532578 IC50 = 2890 nM T16987 CQ0XM6 155532587 Ki = 939.1 nM T16987 CKY1I8 155533416 Ki = 85.5 nM T16987 CDM2Y1 155533454 Ki = 9 nM T16987 C64XYO 155533459 Ki = 5.5 nM T16987 CPX2T1 155533590 Ki = 0.94 nM T16987 COK37H 155533887 Ki > 50000 nM T16987 C3FAC0 155533901 IC50 = 310 nM T16987 C0I5XS 155534055 Ki > 50000 nM T16987 CT5NG1 155534179 Ki = 4.1 nM T16987 CPG13Y 155534247 Ki = 17.6 nM T16987 C6UF3R 155534332 Ki = 8.6 nM T16987 CR2A6J 155534340 Ki = 8.9 nM T16987 C14TGQ 155534675 Ki = 9.3 nM T16987 CK4TR2 155534861 Ki = 76.5 nM T16987 CS5OI9 155534862 Ki = 8.9 nM T16987 CHG10E 155534912 Ki = 10.1 nM T16987 CE1I8S 155535343 Ki = 41.4 nM T16987 CC7M4N 155535347 Ki = 860.7 nM T16987 CVU5P6 155535355 Ki = 39.7 nM T16987 CD2O3A 155535852 Ki = 537 nM T16987 CLJ64Q 155535889 Ki = 13.5 nM T16987 CF0PC4 155536422 Ki = 7 nM T16987 CW92OP 155536652 Ki = 7.7 nM T16987 CB47KF 155536691 Ki = 58.9 nM T16987 CZ0T6A 155537018 Ki = 104.9 nM T16987 C6T7BQ 155537167 Ki = 822 nM T16987 C1K9AC 155537404 Ki = 8965 nM T16987 CXQ23T 155537493 Ki > 100000 nM T16987 C0CG6Q 155537790 Ki = 63.8 nM T16987 C47OHJ 155537809 Ki = 4.6 nM T16987 C67ZET 155537843 Ki = 7.3 nM T16987 C60IZQ 155538189 Ki = 76.8 nM T16987 CB2EI4 155538212 Ki = 36.4 nM T16987 C9AP8F 155538224 Ki = 17.3 nM T16987 CB8C4X 155538289 Ki = 2600 nM T16987 C13GKU 155538478 IC50 = 1600 nM T16987 C3XSM6 155538611 Ki = 837 nM T16987 CM6D1H 155538676 Ki = 7345 nM T16987 CHQP36 155539441 Ki = 19.1 nM T16987 CKE72Y 155539552 Ki = 33.6 nM T16987 C94OZU 155539579 Ki = 2942 nM T16987 CS1G5V 155539783 Ki = 21.3 nM T16987 C53TKA 155540088 Ki = 7.5 nM T16987 CSAD81 155540401 Ki = 46.8 nM T16987 CW9B0X 155540441 Ki = 49.8 nM T16987 C2VAD8 155540596 Ki = 8.2 nM T16987 C95TBC 155540629 Ki > 50000 nM T16987 CCO34J 155540665 Ki = 57.3 nM T16987 CGNS87 155540756 Ki = 9.2 nM T16987 CFN03K 155540920 Ki = 86.3 nM T16987 CGVJ81 155540983 IC50 = 1130 nM T16987 C4H1ZC 155541040 Ki = 32.6 nM T16987 C3CLU2 155541078 Ki = 2.8 nM T16987 C7Z6FC 155541724 Ki = 30.3 nM T16987 C8RV6T 155541805 Ki = 62.3 nM T16987 CW96ES 155541807 Ki = 17.3 nM T16987 C5F3SJ 155541888 Ki = 12.9 nM T16987 CX20DK 155541945 Ki = 2982 nM T16987 CZ2CT0 155542259 Ki = 413 nM T16987 CA75HO 155542580 Ki = 23.8 nM T16987 CTL8O3 155542606 Ki = 7.3 nM T16987 C3RC8T 155542635 Ki = 13.1 nM T16987 CA76LB 155542698 Ki = 790 nM T16987 C2AEH6 155543096 Ki = 804 nM T16987 CHKV89 155543295 Ki = 8.5 nM T16987 CRF64E 155543422 Ki = 9.2 nM T16987 CLF3N5 155543891 Ki = 7.2 nM T16987 CPV20B 155543950 Ki = 26.2 nM T16987 C08DHT 155544006 Ki > 10000 nM T16987 C30HST 155544165 Ki = 10.6 nM T16987 CN0E1V 155544321 Ki = 3.4 nM T16987 CS9WR6 155544336 Ki = 44.5 nM T16987 C7PC5J 155544382 Ki = 9 nM T16987 CSX2H7 155544608 Ki = 59.3 nM T16987 CGP7Z0 155544629 IC50 = 2870 nM T16987 CRM69J 155544710 Ki = 42.6 nM T16987 CP27AW 155544846 Ki = 323.4 nM T16987 CDXL09 155544901 Ki = 7.9 nM T16987 C0BV1J 155545536 Ki = 44.6 nM T16987 CQV78W 155545657 Ki = 9.8 nM T16987 CB6J9G 155545674 Ki > 10000 nM T16987 CP2SZ7 155545812 Ki > 50000 nM T16987 C95IJM 155545916 Ki = 82 nM T16987 CG0E1W 155546684 IC50 = 170 nM T16987 CSW62L 155546892 Ki = 528 nM T16987 CF3UL5 155547275 Ki = 9.5 nM T16987 CV7OB5 155547342 Ki > 100000 nM T16987 C9E2KH 155547486 Ki = 9.5 nM T16987 C59MDT 155547507 Ki = 29.4 nM T16987 C83ZIS 155547526 Ki = 47.2 nM T16987 CW19PC 155547551 Ki = 38.7 nM T16987 C9FVY6 155547723 Ki = 29.5 nM T16987 CK5UD3 155547819 Ki = 43.7 nM T16987 CU94YA 155548070 Ki = 4.7 nM T16987 CCUN29 155548118 Ki = 62.4 nM T16987 C3IO2B 155548134 Ki = 791.7 nM T16987 C3JYG2 155548272 Ki = 744 nM T16987 CQG5F9 155548326 Ki = 39.2 nM T16987 C6XBZ3 155548352 Ki = 35.8 nM T16987 CUTY40 155548640 Ki = 7.8 nM T16987 CH2KB7 155548697 Ki = 8.3 nM T16987 CN7S5W 155548866 Ki = 48.2 nM T16987 CU1NE7 155549031 Ki = 83.4 nM T16987 CR79SY 155549354 Ki = 35.9 nM T16987 CL2B4T 155549378 Ki = 66.4 nM T16987 C6PY2G 155549478 Ki = 20.6 nM T16987 C2CLU0 155549558 Ki = 29.5 nM T16987 CIG6A7 155549616 Ki = 397 nM T16987 C1JR2F 155549662 Ki = 888.3 nM T16987 CF6CW3 155549677 Ki = 83.3 nM T16987 C8NS5F 155549723 Ki = 660 nM T16987 C8GZK4 155549788 Ki > 100000 nM T16987 CAYO49 155550021 Ki = 22.3 nM T16987 C1ZMC2 155550117 IC50 = 250 nM T16987 CZB57Y 155550558 Ki = 8.4 nM T16987 CHO96B 155550610 Ki = 1020 nM T16987 C4O6TN 155550616 Ki = 25.3 nM T16987 CB2Q4M 155550927 Ki = 8.5 nM T16987 CG0MQ3 155551020 Ki = 36 nM T16987 CTE04H 155551088 Ki = 181 nM T16987 CPRC19 155551316 Ki = 91.5 nM T16987 C4S0JZ 155551334 Ki = 47.8 nM T16987 CL2H8V 155551536 Ki = 4600 nM T16987 CSY39H 155551651 Ki = 862 nM T16987 C69AYQ 155551705 Ki > 100000 nM T16987 COC4Z9 155551784 Ki = 15.4 nM T16987 C3AN2K 155551935 Ki = 811 nM T16987 C7E3UF 155552316 Ki = 3600 nM T16987 C3DHB7 155552411 Ki > 50000 nM T16987 CN25FV 155552708 Ki = 1 nM T16987 CBQ42J 155552773 Ki = 550 nM T16987 CFT82G 155552780 Ki = 57.4 nM T16987 CP15VC 155553400 Ki = 58.9 nM T16987 C1QJ3H 155553542 Ki = 74.8 nM T16987 C82WXR 155553544 Ki = 30.1 nM T16987 CQM27S 155553591 Ki = 7.7 nM T16987 CQ1PE4 155553611 Ki > 100000 nM T16987 C02LSY 155553787 Ki = 560 nM T16987 C2J3ZT 155553989 IC50 = 920 nM T16987 C6IMR3 155554140 Ki = 9.8 nM T16987 CMEP40 155554179 Ki = 27.6 nM T16987 CE57CO 155554263 Ki > 50000 nM T16987 C0U8CG 155554286 Ki = 27.2 nM T16987 C6D9BJ 155554303 Ki > 10000 nM T16987 C3W6RT 155554309 Ki > 50000 nM T16987 C7VMB9 155554430 IC50 = 2230 nM T16987 CNX5L2 155554533 Ki = 496.8 nM T16987 C5VLU4 155554670 Ki = 808.9 nM T16987 CM4I0O 155554763 Ki = 650 nM T16987 CW5F4A 155554840 Ki = 196.8 nM T16987 C9W1ET 155555489 Ki = 77 nM T16987 CJ06PN 155555584 Ki > 50000 nM T16987 CV2NZ0 155555718 Ki = 253.2 nM T16987 CUY2C6 155555751 Ki = 8.3 nM T16987 CXNZ49 155555817 Ki = 9.8 nM T16987 CX4P1W 155555874 Ki = 45.3 nM T16987 CWB82E 155555878 Ki = 62.9 nM T16987 CKIR52 155556062 Ki = 9.1 nM T16987 CN9IJ3 155556148 IC50 = 490 nM T16987 C84MNE 155556163 Ki = 23.8 nM T16987 C5PZF2 155556257 Ki = 65 nM T16987 CM60WT 155556386 Ki = 64.3 nM T16987 CD4K6H 155556521 Ki = 8.1 nM T16987 CVR2X5 155556659 Ki > 100000 nM T16987 C2Q3UO 155556889 Ki = 41.9 nM T16987 CYZ3K0 155556908 Ki = 8.2 nM T16987 CG8L0O 155557058 Ki = 921.9 nM T16987 CHKA19 155557282 Ki = 8.7 nM T16987 CRK5I0 155557428 Ki = 89.6 nM T16987 C1RMC6 155557757 Ki = 7.5 nM T16987 CM6NU0 155557925 Ki = 8.1 nM T16987 CWK35T 155557969 Ki = 7.8 nM T16987 CQI5Z4 155558076 Ki = 49.5 nM T16987 CK8GH2 155558119 Ki = 8.2 nM T16987 CME2Z4 155558216 Ki = 39.1 nM T16987 C70WSB 155558230 Ki = 9.7 nM T16987 CQ2ML6 155558561 Ki > 50000 nM T16987 CK1RO0 155558641 Ki = 8.8 nM T16987 C6QXP8 155558748 Ki = 9.4 nM T16987 CI2XS3 155559081 Ki = 26 nM T16987 C6CY3G 155559512 Ki = 9.4 nM T16987 CNT0F5 155559682 Ki = 8.2 nM T16987 CK7H8I 155559761 Ki = 22.9 nM T16987 C3Y7WJ 155560101 Ki = 2000 nM T16987 CZ2A7O 155560148 Ki = 16.8 nM T16987 CB2X0V 155560428 Ki = 8.7 nM T16987 CB5S8V 155560635 Ki = 270.2 nM T16987 COC45S 155560702 Ki = 50.1 nM T16987 CY1TF7 155560798 Ki = 6.3 nM T16987 C0U1NP 155560951 Ki > 50000 nM T16987 CFY9A2 155561027 Ki = 825 nM T16987 CP3H0R 155561119 Ki > 100000 nM T16987 C3FG8W 155561198 Ki = 920 nM T16987 CSK5X2 155561354 Ki = 59.7 nM T16987 C2SZM0 155561361 Ki = 55.1 nM T16987 CY9N4P 155561775 Ki = 78.5 nM T16987 CJ5Y6X 155561851 Ki = 5752 nM T16987 C5W7MQ 155562360 Ki = 51.2 nM T16987 CG43PS 155562766 Ki = 312 nM T16987 C2FW8S 155562815 Ki = 8.3 nM T16987 CJ74ND 155563017 Ki = 35.4 nM T16987 C1J3UH 155563153 Ki > 100000 nM T16987 C7A8EX 155563186 Ki = 26 nM T16987 C9SH6R 155563203 Ki > 100000 nM T16987 C89MTB 155563810 Ki = 767.6 nM T16987 C0GU6P 155563888 Ki = 72.9 nM T16987 CQ40DU 155563908 Ki = 125 nM T16987 C2XB6V 155564028 Ki = 900.8 nM T16987 CF7XH2 155564101 Ki = 93.8 nM T16987 CGY32K 155564210 Ki = 31.8 nM T16987 CY9M4F 155564463 Ki = 8.7 nM T16987 C97TMY 155564559 Ki = 6200 nM T16987 C1K0LR 155564617 Ki = 9.9 nM T16987 CY9IW2 155564942 Ki = 9.8 nM T16987 CNV35X 155565135 Ki = 49.8 nM T16987 C0XO6Z 155565139 Ki = 34.6 nM T16987 C5XV7O 155565283 Ki = 209 nM T16987 CI5MV1 155565395 Ki = 3.6 nM T16987 CJ7I6Z 155565419 Ki = 16.9 nM T16987 CDF5E6 155565628 Ki = 249.1 nM T16987 C0COK6 155565635 Ki = 26.2 nM T16987 CT9Z5H 155565773 Ki > 50000 nM T16987 CW3N9Z 155566095 Ki = 879.2 nM T16987 CD6Z0B 155566206 Ki = 90.1 nM T16987 CCW3L7 155566305 Ki = 459 nM T16987 C5QAM3 155566668 Ki = 33.1 nM T16987 CBV30Y 155566701 Ki = 38.3 nM T16987 CA63FB 155566994 Ki = 52.2 nM T16987 CK80EL 155567119 Ki = 1.3 nM T16987 C4TZ8Q 155567475 Ki = 44.4 nM T16987 CK0M8P 155567487 Ki = 4.4 nM T16987 CL1N9Y 155567612 Ki > 100000 nM T16987 C1MHV5 155567738 Ki = 6538 nM T16987 C29EYS 155567759 Ki = 918.7 nM T16987 CJ2YC4 155567804 Ki = 10.3 nM T16987 CN5OF0 155568108 Ki = 775 nM T16987 CG8QF2 155568247 IC50 = 870 nM T16987 C2ZRJ3 155568270 Ki = 48.6 nM T16987 CDB8T4 155568445 Ki = 59.4 nM T16987 C52NQU 155568453 Ki = 97.1 nM T16987 C35XQY 155568474 Ki = 7.3 nM T16987 CY84TI 155568634 IC50 = 970 nM T16987 C6KR4H 155568759 Ki = 891.9 nM T16987 CQM46K 155568895 IC50 = 540 nM T16987 CH5VU6 155568899 Ki = 33.3 nM T16987 C1C2GI 155569076 Ki = 9.4 nM T16987 CAUR85 155569555 Ki = 760 nM T16987 D00FGB 11414131 Ki = 5.4 nM T16987 D00IAE 11974340 Ki = 8.3 nM T16987 D00IKQ 46703766 Ki = 5.8 nM T16987 D00IUB 13019 Ki = 9200 nM T16987 D00NUK 2837872 Ki = 33 nM T16987 D00RDE 44246261 Ki = 69.4 nM T16987 D00RNZ 910172 Ki = 6500 nM T16987 D00SXO 2793709 Ki = 5.8 nM T16987 D00XIB 11680415 Ki = 0.32 nM T16987 D00XJA 711717 Ki = 6800 nM T16987 D00YEF 148885 Ki = 8.2 nM T16987 D01BUB 94952 Ki = 598000 nM T16987 D01EEM 462919 Ki = 6.4 nM T16987 D01KKU 5281894 Ki = 8400 nM T16987 D01OTW 46703932 Ki = 15.5 nM T16987 D01STY 9861037 Ki = 11 nM T16987 D01UYI 5281607 Ki = 34.7 nM T16987 D01XFH 11851424 Ki = 1 nM T16987 D02BMV 46907399 Ki = 15.6 nM T16987 D02DBP 5054 Ki = 7500 nM T16987 D02JEZ 5281426 Ki = 45.1 nM T16987 D02NQK 46703924 Ki = 13.8 nM T16987 D02QGI 273 Ki = 450 nM T16987 D03APP 4386 Ki = 50 nM T16987 D03DAM 2725651 Ki = 249 nM T16987 D03KRB 45028567 Ki = 4.7 nM T16987 D03NBX 637308 Ki = 8470 nM T16987 D03ZMQ 323 Ki = 8900 nM T16987 D04CVC 4687472 Ki = 1.1 nM T16987 D04HRS 404195 Ki = 5 nM T16987 D04NSN 169682 Ki = 3.2 nM T16987 D04POB 8482 Ki = 49 nM T16987 D04SNH 46933593 Ki = 45.2 nM T16987 D04VSP 46703768 Ki = 5.9 nM T16987 D05EBZ 46703769 Ki = 6.3 nM T16987 D05ETN 46703923 Ki = 6.7 nM T16987 D05JAJ 45028568 Ki = 6.8 nM T16987 D05QOR 5280460 Ki = 4050 nM T16987 D05QUG 45485279 Ki = 7500 nM T16987 D05RAB 45028895 Ki = 28.9 nM T16987 D05TLB 11117301 Ki = 7 nM T16987 D05VVC 44315786 Ki = 3.4 nM T16987 D05WQF 637540 Ki > 1000000 nM T16987 D05XZM 10081162 Ki = 220 nM T16987 D06ALC 6441498 Ki = 4.8 nM T16987 D06DYP 234562 Ki = 5600 nM T16987 D06IOI 901953 Ki = 6.5 nM T16987 D06SZG 44315523 Ki = 7.5 nM T16987 D06XNT 4119643 Ki = 212 nM T16987 D06XVV 64048 Ki = 8650 nM T16987 D06ZMH 2812287 Ki = 10 nM T16987 D06ZOM 15569045 Ki = 593.2 nM T16987 D07AGM 14612854 Ki = 37 nM T16987 D07CYN 20347846 Ki = 1.4 nM T16987 D07LYW 11537386 Ki = 28 nM T16987 D07MTM 403 Ki = 479000 nM T16987 D07PNA 11660633 Ki = 0.69 nM T16987 D07QIU 625902 Ki = 11.2 nM T16987 D07QJJ 289 Ki = 8900 nM T16987 D07TAJ 914298 Ki = 8800 nM T16987 D07UCQ 23680200 Ki = 6250 nM T16987 D07YDN 5281654 Ki = 54.9 nM T16987 D07YSQ 10385283 Ki = 13 nM T16987 D08AIJ 440735 Ki = 31.1 nM T16987 D08AOA 11543564 Ki = 9 nM T16987 D08BFU 5282102 Ki = 4.9 nM T16987 D08JCC 46703770 Ki = 6.9 nM T16987 D09CXX 16122590 Ki = 1340 nM T16987 D09JPC 16402 Ki = 370 nM T16987 D09LUD 4229592 Ki = 13 nM T16987 D09PWX 8739 Ki = 34 nM T16987 D09TES 44395768 Ki = 4.7 nM T16987 D09TKG 25044690 Ki = 16.9 nM T16987 D09USO 5277466 IC50 > 10000 nM T16987 D09WSJ 19772348 Ki = 7.9 nM T16987 D09WVV 8111 Ki = 11400 nM T16987 D0A0YX 5143 Ki = 633 nM T16987 D0A1CM 5281855 Ki = 8150 nM T16987 D0A6HS 6852129 Ki = 3.7 nM T16987 D0A8HW 44395685 Ki = 0.44 nM T16987 D0AU0M 637542 Ki = 8010 nM T16987 D0B5GC 11349 Ki = 6590 nM T16987 D0BD0K 405487 Ki = 7.3 nM T16987 D0C4QB 44395769 Ki = 4.8 nM T16987 D0C7WG 135932620 Ki = 7.3 nM T16987 D0D4OV 20043772 Ki = 7.9 nM T16987 D0D6UR 12394434 Ki = 10500 nM T16987 D0E0RW 69894 Ki = 4140 nM T16987 D0E8CC 18794 Ki = 3.5 nM T16987 D0EJ9B 66827 Ki > 50000 nM T16987 D0F3UR 690836 Ki = 9.9 nM T16987 D0FU0K 23354226 Ki = 5.8 nM T16987 D0G0BJ 51000408 Ki > 50000 nM T16987 D0G0FJ 11206245 Ki = 58 nM T16987 D0G0ZI 403788 Ki > 50000 nM T16987 D0G3BI 25090 Ki = 8000 nM T16987 D0G3TK 5280863 Ki = 145.9 nM T16987 D0G9NE 11659798 Ki = 2.8 nM T16987 D0H3NS 10752 Ki = 2900 nM T16987 D0H4CF 44246267 Ki = 7.3 nM T16987 D0HN0R 11623958 Ki = 9.1 nM T16987 D0IB3K 5320686 Ki = 134.3 nM T16987 D0J2AE 7377 Ki = 125 nM T16987 D0J3SP 11718391 Ki = 2.3 nM T16987 D0J7GU 46703929 Ki = 6.7 nM T16987 D0K3LN 3510137 Ki = 85 nM T16987 D0KB6T 721954 Ki = 21 nM T16987 D0KZ2D 11638641 Ki = 6.2 nM T16987 D0L5TZ 20195365 Ki = 9500 nM T16987 D0L5XK 92249 Ki = 9130 nM T16987 D0LC0F 96876 Ki = 0.39 nM T16987 D0LJ5P 44457221 Ki = 44.5 nM T16987 D0LU4S 156219 Ki = 8600 nM T16987 D0M3PO 69561 Ki = 45 nM T16987 D0M6RM 7365 Ki = 840000 nM T16987 D0M7VN 44392435 Ki = 11 nM T16987 D0M9IQ 23665438 Ki = 5925 nM T16987 D0N1AW 45485270 Ki = 1500 nM T16987 D0N8LR 847760 Ki = 56 nM T16987 D0NN3Q 78105 Ki = 11 nM T16987 D0NS0E 220188 Ki = 104.2 nM T16987 D0O0UE 729977 Ki = 71 nM T16987 D0O4KL 11640067 Ki = 5.5 nM T16987 D0O8WV 11536481 Ki = 5.9 nM T16987 D0OC4B 5357479 Ki = 90.8 nM T16987 D0OI1H 72894 Ki = 0.85 nM T16987 D0OT5L 1631814 Ki = 7600 nM T16987 D0P6AM 3526523 Ki = 20 nM T16987 D0Q0XO 4258082 Ki = 147 nM T16987 D0Q2XB 75928 Ki = 70220 nM T16987 D0Q5VB 46704078 Ki = 8.9 nM T16987 D0Q7DJ 10742 Ki = 9010 nM T16987 D0R4KQ 46704077 Ki = 15.7 nM T16987 D0RB0D 44268050 Ki = 7100 nM T16987 D0RK7J 235259 Ki = 31 nM T16987 D0S0RK 10680 Ki = 7220 nM T16987 D0S2II 308405 Ki = 11.1 nM T16987 D0S9YX 5280373 Ki = 52.5 nM T16987 D0SF3B 11529486 Ki = 52 nM T16987 D0SY2M 5281708 Ki = 56.4 nM T16987 D0T2YZ 3253857 Ki = 138 nM T16987 D0T3NP 7456 Ki = 820 nM T16987 D0TY8X 31036 Ki = 3.4 nM T16987 D0U4BB 10748 Ki = 9700 nM T16987 D0UM1I 12554666 Ki = 10.1 nM T16987 D0V5OW 46907400 Ki = 15.9 nM T16987 D0V9EN 689043 Ki = 9060 nM T16987 D0VD7H 84724 Ki = 33 nM T16987 D0W1AW 4234241 Ki = 835 nM T16987 D0W1OR 7424 Ki = 3670 nM T16987 D0W9VC 670143 Ki = 21 nM T16987 D0X5HL 15107 Ki = 380 nM T16987 D0X6IE 4422372 Ki = 3.5 nM T16987 D0Y3TZ 370 Ki = 7780 nM T16987 D0Y7HG 5281616 Ki = 41.8 nM T16987 D0YD9F 822774 Ki = 68 nM T16987 D0YU8J 1502014 Ki = 3.1 nM T16987 D0YZ5G 5281416 Ki = 9.3 nM T16987 D0Z1HY 67136 Ki = 44 nM T16987 D0ZC3W 6269 Ki = 1.8 nM T97155 D0B3HD 2519 IC50 = 1100000 nM T97155 D06DMQ 59472121 Ki = 0.165 nM T97155 D0H9DA 54761306 IC50 = 4 nM T97155 D0W7HE 56649450 IC50 > 9100 nM T97155 D0XD4I 118502708 IC50 = 6200 nM T97155 D09SFV 3973 IC50 > 10000 nM T97155 CAUK86 108130 IC50 = 7200 nM T97155 CJ19SK 2723790 IC50 = 200 nM T97155 CACS26 11561968 Ki > 10000 nM T97155 CU0E8O 11690457 Ki > 10000 nM T97155 CB0AP2 11705863 Ki > 10000 nM T97155 C1SNR6 13141222 IC50 = 7100 nM T97155 CV9US5 16736978 IC50 > 10000 nM T97155 C0EJK3 23585071 IC50 = 1700 nM T97155 CK2IJ4 25121551 IC50 = 26 nM T97155 C4V2EJ 25261231 IC50 = 4800 nM T97155 CZ3L7W 44233390 IC50 = 41500 nM T97155 CA7R1U 44233391 IC50 = 26200 nM T97155 CH3L9P 44551660 IC50 > 30000 nM T97155 C3VRO9 44557921 IC50 > 5888.44 nM T97155 C28QLM 44605035 IC50 > 50000 nM T97155 C75XHS 44605037 IC50 = 11400 nM T97155 C3F4UX 44605249 IC50 = 7700 nM T97155 CQ0FZ7 44605426 IC50 > 50000 nM T97155 CC7G2L 44605427 IC50 > 50000 nM T97155 CDLP04 44605428 IC50 = 11700 nM T97155 CSKN09 44605429 IC50 > 50000 nM T97155 CA79QG 44605430 IC50 > 50000 nM T97155 CL7C2K 46244173 IC50 = 8 nM T97155 C7D1KH 46244174 IC50 = 8 nM T97155 CE9B8D 46244175 IC50 = 28 nM T97155 C2XN3O 46244255 IC50 = 23 nM T97155 CNI58R 46244256 IC50 = 66 nM T97155 CA26LP 46244257 IC50 = 16 nM T97155 C0YFN7 46244258 IC50 = 15 nM T97155 C2NH0A 46244259 IC50 = 9 nM T97155 CVJM38 46244260 IC50 = 4 nM T97155 CEC3J7 46244352 IC50 = 13 nM T97155 CR40KX 46244453 IC50 = 34 nM T97155 CLZD37 46244883 IC50 = 7 nM T97155 CU5K1G 46834296 IC50 = 620 nM T97155 CM73PR 46834571 IC50 = 1500 nM T97155 CTO5B6 46834572 IC50 = 340 nM T97155 CRJ5W8 51358113 EC50 = 35 nM T97155 CA50HJ 52915004 Ki = 6 nM T97155 C5R2AH 52937148 IC50 = 5200 nM T97155 CLH8Y5 52937149 IC50 = 3000 nM T97155 CT7X9U 52937150 IC50 = 2100 nM T97155 C12GTQ 52937251 IC50 = 180 nM T97155 CQ85UH 52937252 IC50 = 640 nM T97155 CP91TZ 52937253 IC50 = 24 nM T97155 C1MIR4 52937254 IC50 = 130 nM T97155 CID2E8 52937255 IC50 = 1300 nM T97155 C2H9JY 52937257 IC50 = 740 nM T97155 CPY82U 52937258 IC50 = 700 nM T97155 C27QNB 52937357 IC50 = 1400 nM T97155 CFJB79 52937358 IC50 = 400 nM T97155 CT5K9L 52937359 IC50 = 540 nM T97155 C85FTW 52937360 IC50 = 2200 nM T97155 CGLT04 52937361 IC50 = 1600 nM T97155 C2ISM3 52937362 IC50 = 560 nM T97155 C6Q2EN 52937363 IC50 = 180 nM T97155 CFT9H6 52937453 IC50 = 2400 nM T97155 C4C6DF 52937454 IC50 = 1700 nM T97155 C0T8KI 52937455 IC50 = 110 nM T97155 CK30PU 52937456 IC50 = 180 nM T97155 CJU30Y 52937457 IC50 = 1000 nM T97155 C4RJB2 52937458 IC50 = 54 nM T97155 C69SEB 52937459 IC50 = 54 nM T97155 CPR6W2 52937553 IC50 = 26 nM T97155 CQP02L 52937554 IC50 = 12000 nM T97155 CAHU94 52937555 IC50 = 56 nM T97155 CQ2NU7 52937556 IC50 = 1500 nM T97155 CATX20 52937557 Ki = 4 nM T97155 CB9WS5 52937558 IC50 = 2000 nM T97155 CUY01F 52937559 IC50 = 10 nM T97155 CTM68E 52937659 IC50 = 6 nM T97155 C7G9KF 52937660 IC50 = 380 nM T97155 C5G6YD 52937661 IC50 = 460 nM T97155 C6R5OE 52937662 IC50 = 3560 nM T97155 CDHT14 52937663 IC50 = 30 nM T97155 C0IJZ8 52937664 IC50 = 36 nM T97155 CGW25Q 52937665 IC50 = 22 nM T97155 CL04GS 52937759 IC50 = 23 nM T97155 CP0T6S 54761305 IC50 = 240 nM T97155 C0Y9ZG 54761473 IC50 = 6 nM T97155 CZX40J 54761474 IC50 = 23 nM T97155 CT4U1H 54761648 IC50 = 14 nM T97155 C7ONC3 58137106 IC50 = 30 nM T97155 C1YTI8 59472018 Ki = 1 nM T97155 C76CVG 59472034 Ki = 2.4 nM T97155 C1EW0H 59472203 Ki = 0.75 nM T97155 C0MJ3L 59472343 Ki = 0.27 nM T97155 COH62U 60097413 IC50 > 10000 nM T97155 C1MR8Q 60097495 IC50 > 10000 nM T97155 CI1HO0 71521971 Ki = 6 nM T97155 CI2J9Q 71521995 Ki = 90 nM T97155 CKB86I 71537083 Ki = 0.14 nM T97155 CAVL54 71554734 Ki = 4 nM T97155 C70VTD 71557894 Ki = 16 nM T97155 CH45KA 71584052 IC50 = 1500 nM T97155 C6WN9E 71584053 IC50 = 180 nM T97155 C63BLO 71584054 IC50 = 3300 nM T97155 CQ16UM 71584055 IC50 = 3 nM T97155 CS4M6B 71584056 IC50 = 61 nM T97155 C8NLR3 71584161 IC50 = 33 nM T97155 C4UM2I 71584162 IC50 = 46 nM T97155 CN5CK1 71584163 IC50 = 590 nM T97155 C0IMK3 71584164 IC50 = 33 nM T97155 C3QD7S 71584165 IC50 = 360 nM T97155 CAVR57 71584166 IC50 = 1200 nM T97155 CF7H3G 71584281 IC50 = 120 nM T97155 CEH35Y 71584282 IC50 = 130 nM T97155 CZ9SL1 71584283 IC50 = 180 nM T97155 CEN8I0 71584284 IC50 = 14000 nM T97155 CPI9T7 71584285 IC50 > 30000 nM T97155 CW5C4U 71584286 IC50 = 220 nM T97155 CQ2Z9J 71584416 IC50 = 1100 nM T97155 C51YWH 71584417 IC50 = 300 nM T97155 C9LT8N 71584418 IC50 = 24000 nM T97155 C1JHX0 71584419 IC50 = 140 nM T97155 C1V2TU 71584420 IC50 = 41 nM T97155 C51MKU 71584421 IC50 = 4400 nM T97155 CLO1P5 72199292 IC50 = 14 nM T97155 C0V8OG 86306050 IC50 = 0.5 nM T97155 CHX2Z3 90435584 Ki = 0.21 nM T97155 CL3MG7 117906028 IC50 = 180 nM T97155 C53UXY 118025505 IC50 = 158 nM T97155 CM3JO2 118025835 IC50 = 1860 nM T97155 CC1FP6 118025908 IC50 = 654 nM T97155 C5TQU3 118025943 IC50 = 3560 nM T97155 C05LQH 118498627 IC50 > 30000 nM T97155 CXCF46 118498683 IC50 > 30000 nM T97155 CJA07S 118498727 IC50 = 4400 nM T97155 CG6D1J 118498935 IC50 > 30000 nM T97155 CXR46C 118499887 IC50 > 30000 nM T97155 CFVN15 118500050 IC50 > 30000 nM T97155 CY9NW0 118500097 IC50 > 24000 nM T97155 CXEI18 118500108 IC50 > 30000 nM T97155 CL2Z5Y 118502821 IC50 > 30000 nM T97155 CVY64N 118502892 IC50 > 30000 nM T97155 CO20ET 118502895 IC50 > 2600 nM T97155 CU1X3H 118502919 IC50 > 23000 nM T97155 CRAF61 118523357 IC50 > 24000 nM T97155 C5P7VH 118523411 IC50 > 30000 nM T97155 CD0EY5 118523423 IC50 > 29000 nM T97155 CQX38N 118720611 IC50 = 0.5 nM T97155 CFP58Q 118720612 IC50 = 1 nM T97155 CF5HV8 118720613 IC50 = 0.3 nM T97155 C2UIB7 118720614 IC50 = 1 nM T97155 CSH50J 118720615 IC50 = 0.4 nM T97155 C4BD5I 118720616 IC50 = 29 nM T97155 C08TCW 118720617 IC50 = 2 nM T97155 C1BHL8 118720618 IC50 = 440 nM T97155 CW3FG8 118720619 IC50 = 6200 nM T97155 CA8YI7 118720620 IC50 = 2100 nM T97155 CBIK65 118720621 IC50 = 41 nM T97155 C0PYH3 118720622 IC50 = 64 nM T97155 CVIT16 118720879 IC50 = 96 nM T97155 CJW06C 118720880 IC50 = 95 nM T97155 C1R3VQ 118720881 IC50 = 39 nM T97155 C86RWG 118720882 IC50 = 26 nM T97155 CYSD60 118720883 IC50 = 5 nM T97155 C6E9UN 118720884 IC50 = 1 nM T97155 C4LW6I 118720885 IC50 = 0.2 nM T97155 C9Y4EH 118720886 IC50 = 0.4 nM T97155 C5Q2ZW 118720887 IC50 = 0.1 nM T97155 CMTR04 118720888 IC50 = 34 nM T97155 CMP6U7 118720889 IC50 = 6 nM T97155 CFUA64 118720890 IC50 = 190 nM T97155 C9SF2E 118720891 IC50 = 0.5 nM T97155 CK68CA 130453737 IC50 > 30000 nM T97155 CDP9S1 130470501 IC50 > 30000 nM T97155 C5U1XV 130470509 IC50 > 30000 nM T97155 CLTQ15 130470516 IC50 > 25000 nM T97155 CUO41K 130470684 IC50 > 19000 nM T97155 CPC2A7 130470749 IC50 > 30000 nM T97155 C7QI1J 131986481 IC50 = 10000 nM T97155 CV97TQ 132167490 IC50 < 10 nM T97155 C28LIU 132178541 IC50 < 10 nM T97155 CX7I1W 132178548 IC50 = 10 nM T97155 CR4MH7 132178746 IC50 = 10 nM T97155 C4T6FV 132179226 IC50 = 10 nM T97155 C4Z6CL 132179249 IC50 = 10 nM T97155 CSWE45 134163712 IC50 = 87 nM T97155 CX0UR7 134694318 IC50 > 30000 nM T97155 C9FUK2 135151360 IC50 > 29000 nM T97155 C81NTE 135980524 IC50 = 2400 nM T97155 C0AYN4 135980525 IC50 = 320 nM T97155 C0EY8G 138490470 IC50 > 30000 nM T97155 CQ2M5F 138504490 IC50 > 30000 nM T97155 CKDZ26 138504497 IC50 > 30000 nM T97155 CH2D8T 145949518 IC50 > 30000 nM T97155 C9Q1TH 145950015 IC50 > 30000 nM T97155 CK64FQ 145950570 IC50 > 30000 nM T97155 C6JYA5 145950619 IC50 = 3100 nM T97155 CPE7N3 145950719 IC50 > 30000 nM T97155 CW6XJ2 145951187 IC50 > 16000 nM T97155 CCOW60 145952011 IC50 > 26000 nM T97155 CVR31U 145952361 IC50 > 30000 nM T97155 C2WFH6 145953847 IC50 > 13000 nM T97155 CTRQ36 145954357 IC50 > 28000 nM T97155 CN7T2Q 145954771 IC50 > 30000 nM T97155 CHR53Q 145957373 IC50 > 27600 nM T97155 C6R0OC 145957812 IC50 > 30000 nM T97155 CA4C9J 145957925 IC50 > 30000 nM T97155 C73CBD 145959061 IC50 = 15000 nM T97155 C75LGW 145959260 IC50 = 2000 nM T97155 CS13IP 145959347 IC50 = 51 nM T97155 CDYO54 145959735 IC50 > 20000 nM T97155 C14WSR 145963769 IC50 = 580 nM T97155 CS2KD5 145963991 IC50 > 30000 nM T97155 CHRZ36 145964774 IC50 > 30000 nM T97155 C6BQY4 145964941 IC50 > 30000 nM T97155 C1I5GU 145964978 IC50 > 30000 nM T97155 C8CS7N 145965459 IC50 = 4620 nM T97155 C8K3NI 145965633 IC50 = 1590 nM T97155 CJ1R2W 145965788 IC50 > 30000 nM T97155 CCZ6K5 145966304 IC50 > 30000 nM T97155 C9PA0X 145966721 IC50 > 30000 nM T97155 C9C7KV 145966818 IC50 = 22400 nM T97155 C9MB3A 145967469 IC50 > 30000 nM T97155 CD71MG 145968213 IC50 > 30000 nM T97155 C5K0LN 145969815 IC50 > 30000 nM T97155 CZNQ73 145971262 IC50 > 30000 nM T97155 C9R2VH 145971456 IC50 > 30000 nM T97155 CIF4D8 145971589 IC50 = 1320 nM T97155 CVC90R 145971640 IC50 > 30000 nM T97155 C54YDF 145972329 IC50 = 19100 nM T97155 CRTG91 145973095 IC50 > 30000 nM T97155 CA7X9N 145973949 IC50 = 2630 nM T97155 CN0EB3 145974305 IC50 > 30000 nM T97155 C5DIA6 145976562 IC50 = 19300 nM T97155 C07XEP 145977110 IC50 > 30000 nM T97155 CP67AD 145977670 IC50 = 66 nM T97155 CA93IU 145977679 IC50 = 269 nM T97155 CDM3E8 145978228 IC50 > 30000 nM T97155 C1B6FV 145978350 IC50 > 30000 nM T97155 CU21SN 145979565 IC50 = 5100 nM T97155 CVAQ91 145979907 IC50 = 130 nM T97155 C2C3LB 145980103 IC50 = 270 nM T97155 CT8I7V 145980208 IC50 = 550 nM T97155 CG9C1M 145980501 IC50 = 5 nM T97155 CGA83C 145981271 IC50 = 2 nM T97155 C0JU1P 145981505 IC50 = 37 nM T97155 CSJ3P8 145983402 IC50 = 17 nM T97155 CN4D6T 145986333 IC50 = 360 nM T97155 C5R6BS 145987142 IC50 = 2 nM T97155 C8T1NP 145987199 IC50 = 4000 nM T97155 C7KVT0 145987381 IC50 = 51 nM T97155 CDBT65 145989852 IC50 = 260 nM T97155 C60ZFB 145990007 IC50 = 2 nM T97155 CP84US 145990234 IC50 = 100 nM T97155 CEO1F8 145991167 IC50 = 21 nM T97155 C7B2KM 145991457 IC50 = 11 nM T97155 CYO9J4 145991697 IC50 = 17 nM T97155 C2J0XO 145992074 IC50 = 15 nM T97155 C0HO8J 145992301 IC50 = 18 nM T97155 C7E9MS 145992816 IC50 = 86 nM T97155 CI1YX3 145993592 IC50 = 8 nM T97155 C8X2IT 145996536 IC50 = 394 nM T97155 C9UF6S 155510524 IC50 > 30000 nM T97155 CH8J7L 155510809 Ki = 1 nM T97155 COM30P 155514391 Ki = 1 nM T97155 CY1B4L 155517765 Ki = 5 nM T97155 CSPN68 155532569 Ki = 1.24 nM T97155 C23IEP 155536557 Ki = 21 nM T97155 CG15CZ 155539194 IC50 = 3200 nM T97155 C13HGT 155541849 IC50 > 30000 nM T97155 CKIJ48 155543371 IC50 > 30000 nM T97155 CG7D9R 155543873 IC50 = 5500 nM T97155 CBN29V 155544583 IC50 = 4700 nM T97155 CW9F7M 155544669 IC50 > 30000 nM T97155 CHCS54 155546044 Ki = 2 nM T97155 C6KXY5 155546286 IC50 = 11000 nM T97155 CPK82D 155546294 IC50 > 30000 nM T97155 CU2QO9 155547462 IC50 > 30000 nM T97155 CY6F3D 155547951 IC50 = 2600 nM T97155 CG8FO4 155548512 IC50 > 30000 nM T97155 C8JI1D 155550286 IC50 = 7100 nM T97155 CQ5OD0 155550395 IC50 = 1900 nM T97155 CAJ57R 155550406 IC50 > 30000 nM T97155 CR8DO6 155550599 IC50 = 3000 nM T97155 C5LTO0 155551695 IC50 = 730 nM T97155 CJL9K4 155552042 IC50 > 30000 nM T97155 CJ75BO 155552100 IC50 = 8500 nM T97155 CX6QO1 155552713 IC50 > 11000 nM T97155 C2ZNL8 155552880 IC50 = 3500 nM T97155 C09TOV 155553799 IC50 > 14000 nM T97155 CHP3R7 155554099 IC50 > 30000 nM T97155 C0I4KF 155555078 IC50 > 30000 nM T97155 CS8C4B 155555411 IC50 > 18000 nM T97155 C92NTS 155558433 IC50 > 30000 nM T97155 CAV79P 155560264 IC50 > 30000 nM T97155 CO3R8Y 155560892 Ki = 0.53 nM T97155 C9UYA8 155561280 IC50 > 23000 nM T97155 CH9UY6 155562079 IC50 > 30000 nM T97155 CP52DQ 155562348 IC50 > 18000 nM T97155 CG9QR6 155563968 IC50 > 30000 nM T97155 CB7SJ5 155564720 IC50 = 1200 nM T97155 CXKI62 155567017 IC50 > 15000 nM T97155 C7KPT9 155567536 IC50 > 13000 nM T97155 C8INK5 155568740 IC50 = 640 nM T97155 C1S8ZB 155568922 IC50 = 4400 nM T97155 CQR7E9 155569091 IC50 > 30000 nM T97155 CE6P9C 155569571 Ki = 26 nM T97155 D00PXO 6605258 IC50 = 200 nM T97155 D02TSN 46244454 IC50 = 5 nM T97155 D03EHM 24905142 IC50 = 1420 nM T97155 D05USL 5278396 IC50 > 30000 nM T97155 D0G0BJ 51000408 IC50 = 26 nM T97155 D0R0TW 11964036 IC50 > 10000 nM T97155 D0T0BY 10039361 IC50 > 100000 nM T97155 D0U8YN 398148 IC50 = 6700 nM T97155 D0W1ST 9860529 IC50 > 100000 nM T97155 D0X7TB 10017389 IC50 > 100000 nM T97155 D0Y3OO 11327430 IC50 > 10000 nM T30414 CTZ6A9 748659 IC50 = 785 nM T30414 C98PBF 752812 IC50 = 140 nM T30414 CUA0F3 71148609 IC50 = 793 nM T30414 CX9V0U 71148612 IC50 = 646 nM T30414 CI01TH 71148620 IC50 = 5130 nM T30414 C5T8ZC 71148622 IC50 = 336 nM T30414 C7R1WH 71769562 IC50 = 0.0043 nM T30414 CTX46Q 71770951 IC50 = 2.4 nM T30414 C83GPX 72201708 IC50 = 1600 nM T30414 C5PVQ8 72201854 IC50 = 24 nM T30414 C6UX9C 72203403 IC50 = 270 nM T30414 C7SKI2 89873469 IC50 = 1.69 nM T30414 C1DZ9W 89873480 IC50 = 2.8 nM T30414 CD6YU8 89873584 IC50 = 1800 nM T30414 CB6I1D 89880942 IC50 = 0.98 nM T30414 CQ68FB 89880953 IC50 = 37 nM T30414 CP6Z1H 89880954 IC50 = 38 nM T30414 CHX28P 89880970 IC50 = 110 nM T30414 CP3TV0 89881055 IC50 = 3.1 nM T30414 CEF4R0 89881089 IC50 = 530 nM T30414 C24JRI 118068374 IC50 = 7.6 nM T30414 C0VUO7 118068383 IC50 = 1.3 nM T30414 C2LPS6 118068437 IC50 = 1.2 nM T30414 CYP8Z0 118068442 IC50 = 0.99 nM T30414 CIU52M 118068455 IC50 = 220 nM T30414 C8B7QI 118068465 IC50 = 26 nM T30414 CU6G9K 118068468 IC50 = 2100 nM T30414 CE3N8D 118070586 IC50 = 2900 nM T30414 CPO5E7 118070587 IC50 = 67 nM T30414 C4OVE8 118714099 IC50 = 66 nM T30414 CSQO76 118714113 IC50 > 10000 nM T30414 C2GC9I 118714140 IC50 = 10000 nM T30414 C57IKA 118714146 IC50 = 279 nM T30414 CC4LA1 118953461 IC50 = 132 nM T30414 CY6RC8 118953471 IC50 > 10000 nM T30414 CB14QU 118967085 IC50 = 2187.76 nM T30414 C2J6CW 118967088 IC50 > 10000 nM T30414 C13EIL 118967091 IC50 = 450 nM T30414 C0QC6B 118967102 IC50 > 10000 nM T30414 CT2NJ6 118967103 IC50 > 10000 nM T30414 C8GFK0 118967104 IC50 > 10000 nM T30414 C5OKW0 118967130 IC50 = 5110 nM T30414 C69BXT 118967132 IC50 = 4786.3 nM T30414 CKXI20 118971050 IC50 = 3715.35 nM T30414 C2GHX9 118971053 IC50 > 10000 nM T30414 C51GPE 118971054 IC50 = 1380.38 nM T30414 CE3CN6 118971057 IC50 = 489.78 nM T30414 C7W8EF 118971059 IC50 = 4897.79 nM T30414 CT4RP7 118971061 IC50 = 204.17 nM T30414 CU5CI9 118971160 IC50 > 10000 nM T30414 C0VB7P 118971189 IC50 > 10000 nM T30414 COY4L9 118971366 IC50 = 1350 nM T30414 CD7AN0 118971371 IC50 = 812.83 nM T30414 C2Z3QP 118971373 IC50 = 1500 nM T30414 C17AOH 118971381 IC50 = 4150 nM T30414 CW03MF 126961335 IC50 = 380 nM T30414 CYDW03 132051219 IC50 = 36.3 nM T30414 C7JEQ8 132051220 IC50 = 1318.26 nM T30414 CBU5Z8 132051221 IC50 = 15.49 nM T30414 CNZ8G5 132051226 IC50 = 4786.3 nM T30414 C42CAO 132051227 IC50 < 10000 nM T30414 C0L2AM 132051232 IC50 = 588.84 nM T30414 C4WR7C 132051234 IC50 = 57.2 nM T30414 C1LP5I 132051237 IC50 = 39.5 nM T30414 CLS13X 132051238 IC50 = 28.18 nM T30414 CLNR21 132051239 IC50 = 436.52 nM T30414 CGR58D 132051241 IC50 > 10000 nM T30414 CV0P3B 132051242 IC50 = 1200 nM T30414 C7EUD6 132051243 IC50 = 933.25 nM T30414 C7G5QV 132051298 IC50 = 1090 nM T30414 CB60QN 132051300 IC50 = 1288.25 nM T30414 CU26YD 132051301 IC50 = 173.78 nM T30414 C2BN5A 132051302 IC50 = 757 nM T30414 CL3PT6 132051307 IC50 = 207 nM T30414 CC5X0I 132051309 IC50 = 675 nM T30414 CTA7C8 132051310 IC50 = 2511.89 nM T30414 COX1G5 132051312 IC50 < 10000 nM T30414 CWRT29 132051314 IC50 = 352 nM T30414 CHO8A9 132051315 IC50 = 524.81 nM T30414 COJ98T 132051319 IC50 = 52.3 nM T30414 C28YUC 132051372 IC50 = 406 nM T30414 CJ1Q3F 134134975 IC50 > 10000 nM T30414 C3W6CY 134135549 IC50 = 3400 nM T30414 CUO21P 134137936 IC50 = 19.95 nM T30414 C5IE4P 140928469 IC50 > 10000 nM T30414 C7ZXS6 145998086 IC50 = 820 nM T30414 C1GBW0 147630030 IC50 = 3.3 nM T30414 C0T6JE 155511382 IC50 = 1900 nM T30414 C2H6XF 155515625 IC50 = 2.4 nM T30414 CY9P7W 155517852 IC50 = 19 nM T30414 C3QH4N 155521862 IC50 = 1.6 nM T30414 CRH6N2 155523135 IC50 = 4.3 nM T30414 C3BP0C 155523812 IC50 = 11 nM T30414 CVR28C 155525561 IC50 = 1.1 nM T30414 CCS17U 155527266 IC50 = 9.4 nM T30414 C6XR4F 155528420 IC50 = 1.2 nM T30414 C8UGH9 155529126 IC50 = 410 nM T30414 C47BZM 155530857 IC50 = 3.2 nM T30414 CEN25I 155538309 IC50 = 3.4 nM T30414 CUX8T6 155543857 IC50 = 3.1 nM T30414 CW9R1G 155544936 IC50 = 3.2 nM T30414 CMPU79 155545221 IC50 = 27 nM T30414 C6HJK0 155548776 IC50 = 2.3 nM T30414 CQT80A 155549758 IC50 = 1.6 nM T30414 CR5FT2 155555810 IC50 = 0.81 nM T30414 CK5U6H 155563531 IC50 = 760 nM T30414 C1E2JR 155565675 IC50 = 1.8 nM T30414 D00KRL 10132921 IC50 = 130 nM T86350 D07POC 176870 IC50 = 10 nM T86350 D0O8GK 71496458 IC50 = 2.1 nM T86350 D0BM7M 11488320 IC50 = 4 nM T86350 D0M4AV 57335384 IC50 = 46 nM T86350 D0R0LB 91668194 IC50 = 4 nM T86350 CX17CH 701322 IC50 = 96 nM T86350 C5MI4N 14246200 IC50 = 45300 nM T86350 C5SYC3 67304928 IC50 > 10000 nM T86350 CSM8Q3 71524871 IC50 = 55600 nM T86350 CQ34CK 71524919 IC50 = 40200 nM T86350 CZQ2S4 71524965 IC50 = 63200 nM T86350 C8A9IN 71525006 IC50 = 51700 nM T86350 C0M4LC 71525009 IC50 = 35900 nM T86350 C1D3KG 71535003 IC50 = 21 nM T86350 CM1VR8 74766099 IC50 = 1 nM T86350 C78NRU 112865697 IC50 = 230 nM T86350 CI6H8C 112865788 IC50 = 1573 nM T86350 COU61I 112865858 IC50 > 10000 nM T86350 CIR97O 112866175 IC50 = 18 nM T86350 C2BAR8 112866205 IC50 = 1745 nM T86350 CKX0H7 118073560 IC50 = 2 nM T86350 CGT4R5 118073677 IC50 = 2 nM T86350 CLQO21 118073729 IC50 = 9 nM T86350 CCXT19 141510925 IC50 = 2 nM T86350 C9ED8K 141510928 IC50 = 1.7 nM T86350 C7TW9O 141510929 IC50 = 1.2 nM T86350 COLJ50 141510933 IC50 = 1.9 nM T86350 C0AU5J 141510934 IC50 = 2.6 nM T86350 CI5KY6 141510937 IC50 = 5.8 nM T86350 C06YIS 145968559 IC50 = 4.2 nM T86350 CVXS26 145969908 IC50 = 2.4 nM T86350 C0XH6S 145970573 IC50 = 4.2 nM T86350 CG57KO 145977147 IC50 = 36 nM T86350 CCT8N6 145978865 IC50 = 167 nM T86350 C5LIK2 145980611 IC50 = 1608 nM T86350 C1A5PW 145980662 IC50 = 21 nM T86350 C8FRT3 145981115 IC50 > 10000 nM T86350 C4J9SC 145981182 IC50 = 183 nM T86350 CP67EO 145981349 IC50 > 10000 nM T86350 CPHN84 145985403 IC50 = 619 nM T86350 CV45JH 145986520 IC50 = 1209 nM T86350 CU96RK 145987761 IC50 = 1322 nM T86350 C0MI7K 145988025 IC50 = 69 nM T86350 C3N8OJ 145988373 IC50 = 167 nM T86350 CE1QB4 145990507 IC50 = 236 nM T86350 CNQ91H 145990537 IC50 = 60 nM T86350 CZP7Y0 145992597 IC50 = 1847 nM T86350 C4A2UC 145992646 IC50 > 10000 nM T86350 CO41PW 145992706 IC50 = 825 nM T86350 C0C4ZD 145993006 IC50 = 27 nM T86350 C7Q6NU 145993198 IC50 = 1345 nM T86350 CZ6OC9 145993414 IC50 = 31 nM T14252 D0ED7U 60648 IC50 = 917000 nM T14252 D08ESA 198693 IC50 = 333000 nM T14252 D0C9XA 119 IC50 = 1000 nM T14252 CJ9V4G 40598 IC50 > 1000000 nM T14252 CXSD61 155246 IC50 = 43700 nM T14252 CHV0G9 639062 IC50 > 1000000 nM T14252 C97FYX 702501 IC50 > 300000 nM T14252 C8X9TQ 1069892 Ki > 100000 nM T14252 C1A0UL 1502074 IC50 = 2300 nM T14252 C3DR8J 1502075 IC50 = 2511.89 nM T14252 C9EI4M 1530639 IC50 > 1000000 nM T14252 CU23IC 4531494 IC50 = 10000 nM T14252 CG1ZF6 5311322 Ki = 6100 nM T14252 CN2C7Q 6604883 IC50 = 86000 nM T14252 C4A6SU 8181355 IC50 > 500000 nM T14252 CQ64IH 9797818 IC50 = 1990000 nM T14252 C31HNE 9884272 Ki > 100000 nM T14252 CY2IS7 9888224 IC50 = 46000 nM T14252 CI06JL 9982662 IC50 = 198000 nM T14252 CTZ5Q7 9983570 IC50 = 1080000 nM T14252 C75BDY 10031163 IC50 = 212000 nM T14252 CZ4PO2 10050339 IC50 = 6740000 nM T14252 CZQ52G 10052359 IC50 = 169000 nM T14252 CP2WF1 10072112 IC50 = 142000 nM T14252 CG1A4H 10073933 IC50 = 25000 nM T14252 C57RVK 10075407 IC50 = 142000 nM T14252 C4S1CO 10096504 IC50 = 25000 nM T14252 CXJR61 10252950 IC50 = 178000 nM T14252 CC8V4E 10412575 IC50 = 20000 nM T14252 CZ8FQ2 10481573 IC50 = 29000 nM T14252 CU40KP 11743493 IC50 = 91000 nM T14252 CH6GX1 13314232 IC50 > 500000 nM T14252 C03OAI 14810154 IC50 = 8128.31 nM T14252 C6VK4E 17173775 IC50 > 1000000 nM T14252 CE92MX 17174058 IC50 > 1000000 nM T14252 C3OQD7 17250318 IC50 > 500000 nM T14252 CME93B 43345728 IC50 > 1000000 nM T14252 C5JUW9 47058964 IC50 > 1000000 nM T14252 CLIK30 50941729 IC50 > 100000 nM T14252 CQ4XJ7 55285849 IC50 = 13900 nM T14252 CY9O8W 55285850 IC50 = 13900 nM T14252 C8UTR2 67642717 IC50 = 1900 nM T14252 C6ME5H 70684991 IC50 = 876000 nM T14252 C79CYX 70689234 IC50 = 2043000 nM T14252 CD9EV5 70691307 IC50 = 782000 nM T14252 CJ7P8C 70691309 IC50 = 3233000 nM T14252 C53QGB 118711599 IC50 = 76300 nM T14252 CO18BS 137635197 IC50 = 405000 nM T14252 CQL64H 137637846 IC50 > 1000000 nM T14252 CZ73DV 137638595 IC50 > 100000 nM T14252 CARI53 137638617 IC50 > 100000 nM T14252 CUM2T0 137638836 IC50 > 100000 nM T14252 C3PY5G 137638838 IC50 > 50000 nM T14252 CP7OV5 137639241 IC50 > 100000 nM T14252 C21IZT 137639281 IC50 > 1000000 nM T14252 CP24OX 137642163 IC50 > 100000 nM T14252 CK2VU3 137650102 IC50 > 1000000 nM T14252 C52PYO 137650910 IC50 > 1000000 nM T14252 CS6FX4 137651374 IC50 > 1000000 nM T14252 CPLJ94 137651669 IC50 > 1000000 nM T14252 CN04QK 137652511 IC50 > 1000000 nM T14252 CGC1Z4 137654858 IC50 > 50000 nM T14252 CADN74 137657292 IC50 > 100000 nM T14252 C4NK1W 137658990 IC50 > 50000 nM T14252 CPI4S8 137659917 IC50 > 50000 nM T14252 CI7S8H 155516242 IC50 > 100000 nM T14252 CL2TZ4 155518880 IC50 = 2754.23 nM T14252 C4U8QT 155524561 IC50 > 100000 nM T14252 CJ4OV6 155530359 IC50 > 100000 nM T14252 C4RL9X 155535776 IC50 > 100000 nM T14252 C7XS6Z 155549186 IC50 = 9332.54 nM T14252 CL2Q6G 155567178 IC50 > 100000 nM T14252 D02ANG 5216267 IC50 = 125892.54 nM T14252 D03IWW 6575389 IC50 = 2320000 nM T14252 D08YGM 92409 IC50 = 944000 nM T14252 D0D2EF 1796510 IC50 = 51000 nM T14252 D0H7WK 10458835 IC50 = 5000 nM T14252 D0P3KI 9888030 IC50 = 8920 nM T14252 D0RF2M 4498 IC50 = 106000 nM T14252 D0V5OY 16725912 Ki > 100000 nM T14252 D0V7RG 3532 IC50 = 110000 nM T14252 D0W8SX 239 IC50 = 41200 nM T14252 D0X3CF 442879 IC50 > 500000 nM T07173 D03ZBT 11626560 IC50 < 1 nM T07173 D04LVK 57379345 IC50 = 2727 nM T07173 D07TOK 46188928 IC50 = 2 nM T07173 D0AF6O 71731823 IC50 = 24 nM T07173 D0OB0F 5328940 IC50 = 22 nM T07173 D0Y5UG 2160 EC50 = 86000 nM T07173 D00DRL 44137946 IC50 = 46 nM T07173 D01HKZ 57345941 IC50 < 3 nM T07173 D02QWY 24785538 IC50 = 7 nM T07173 D02RJY 11442891 IC50 = 30 nM T07173 D03HUX 49792852 IC50 > 10000 nM T07173 D03QLG 9917013 IC50 > 10000 nM T07173 D03UDF 129103609 IC50 = 0.98 nM T07173 D05NFR 135565923 IC50 = 0.4 nM T07173 D08QGT 17755052 IC50 = 2850 nM T07173 D0E3TC 44259 IC50 = 1.7 nM T07173 D0FA6S 54576299 IC50 = 0.85 nM T07173 D0FD6D 11751922 IC50 = 3 nM T07173 D0MP0X 16659841 IC50 = 3 nM T07173 D0O0LS 25141092 IC50 = 2.9 nM T07173 D0O6WV 24794418 IC50 = 290 nM T07173 D0P1CV 46191454 IC50 > 10000 nM T07173 D0Q9UX 16718576 IC50 = 53 nM T07173 D0WS1V 448991 IC50 = 1710 nM T07173 D05NBR 74220979 IC50 < 100 nM T07173 D0BP9B 90168931 IC50 < 100 nM T07173 D0JU4R 73891136 IC50 < 100 nM T07173 D0H4GI 10275001 IC50 > 3000 nM T07173 D0T3ME 156422 IC50 = 160 nM T07173 C1ZG2U 449087 IC50 > 10000 nM T07173 C18WEB 490561 IC50 = 13 nM T07173 CR5X9Q 707935 IC50 = 27 nM T07173 COH21C 951145 IC50 = 303 nM T07173 CU9J0H 2125863 IC50 = 2.7 nM T07173 CA0X4D 2434227 IC50 = 5000 nM T07173 CO84PB 2455929 IC50 = 5000 nM T07173 CY9D7W 2517470 IC50 = 143.7 nM T07173 CVL95J 2535914 IC50 = 137 nM T07173 CJ59NC 2541025 IC50 = 1017.1 nM T07173 C2XRI8 2547426 IC50 = 5000 nM T07173 C7UN1Z 2597009 IC50 = 121.7 nM T07173 CF89XO 2597103 IC50 = 259.6 nM T07173 CCE6F2 2826530 IC50 = 5880 nM T07173 CXVB08 3399504 IC50 = 667.7 nM T07173 CJ3Q5R 3666186 IC50 = 50 nM T07173 CJM9Q8 4410298 IC50 = 53.6 nM T07173 CV1PK6 4798875 IC50 = 77.6 nM T07173 CJU3B9 4798877 IC50 = 371.4 nM T07173 C5AW4U 4802531 IC50 = 773.5 nM T07173 CR1HA0 4802711 IC50 = 97.4 nM T07173 C9QD7T 4802738 IC50 = 5000 nM T07173 C1DW3F 5019229 IC50 = 283.5 nM T07173 CPZY43 5121984 IC50 = 3300 nM T07173 C7WO8K 7190453 IC50 = 204.6 nM T07173 C7SCJ2 9206007 IC50 = 1424 nM T07173 CK21EQ 9796713 IC50 = 162 nM T07173 CJR93U 9809634 IC50 > 1000 nM T07173 CSQ85J 9827373 IC50 = 8 nM T07173 CJH69P 9840393 IC50 = 88 nM T07173 CH3QK5 9852367 IC50 > 1000 nM T07173 C4R0JM 9874223 IC50 > 1000 nM T07173 CE7BQ0 9874626 IC50 > 1000 nM T07173 CWT83F 9885305 IC50 = 47000 nM T07173 C3RL6K 9890129 IC50 = 2.9 nM T07173 CRO5D3 9912410 IC50 = 5 nM T07173 CU7QI4 9937567 IC50 = 270 nM T07173 CAM14L 9938261 IC50 = 210 nM T07173 CR3DA5 9939328 IC50 > 10000 nM T07173 C61KBJ 9943464 IC50 = 12 nM T07173 CA96JS 9999629 IC50 = 344 nM T07173 CVBH40 9999630 IC50 = 28 nM T07173 CUJR40 10062694 EC50 > 2000 nM T07173 C3A5GM 10157542 IC50 = 65 nM T07173 C59FGN 10165455 IC50 = 1 nM T07173 C9J2KW 10181704 IC50 = 240 nM T07173 C07ULE 10226065 IC50 = 80 nM T07173 CSGD16 10246246 IC50 > 7000 nM T07173 CG8K7O 10248990 IC50 = 19 nM T07173 CJB8K3 10275928 IC50 = 1100 nM T07173 C64JPR 10301519 IC50 = 50 nM T07173 C7P1OA 10341317 IC50 = 179 nM T07173 CAJ43D 10422105 IC50 = 55800 nM T07173 C7HBP6 10429593 IC50 > 10000 nM T07173 C8J9NC 10429704 IC50 = 47 nM T07173 CRJD61 10532168 IC50 > 1000 nM T07173 CHB35P 10604501 IC50 > 1000 nM T07173 C05KFQ 10604778 IC50 > 1000 nM T07173 CJ4BN2 10626594 IC50 = 270 nM T07173 CGP93J 10745853 IC50 = 210 nM T07173 CO7Y9M 10770450 IC50 > 10000 nM T07173 CJ67CS 11212221 EC50 = 6 nM T07173 CWC2X6 11223992 IC50 = 20 nM T07173 C3QKJ0 11281671 IC50 = 3 nM T07173 CBOP58 11293798 Ki > 10000 nM T07173 C26BZX 11362471 Ki > 10000 nM T07173 CWXB93 11397177 Ki > 10000 nM T07173 CF1L3B 11441796 IC50 = 15 nM T07173 C2T8YD 11511361 IC50 = 500 nM T07173 C1A7EI 11524587 IC50 = 160 nM T07173 CTG83F 11539329 Ki > 2500 nM T07173 C6YU9Z 11560696 IC50 = 120 nM T07173 CMIL86 11590363 Ki > 2500 nM T07173 C4U7HM 11621097 IC50 = 7 nM T07173 CZ4F7B 11621437 IC50 > 1000 nM T07173 CYL45U 11634544 IC50 = 19 nM T07173 C9T6SC 11640926 Ki > 2500 nM T07173 CQ4OC2 11654378 IC50 = 11 nM T07173 C36EVF 11705812 IC50 = 7 nM T07173 C45EWD 11723489 IC50 > 7000 nM T07173 CGY1R0 11740295 IC50 = 33 nM T07173 CQ3N4E 11756662 IC50 = 4000 nM T07173 C4NO7Y 11809063 IC50 = 155 nM T07173 C9JT4S 11847343 IC50 = 181 nM T07173 CJE7O8 11952607 IC50 = 34.3 nM T07173 C16CKR 11978342 EC50 = 4 nM T07173 CR1ZQ8 11978448 EC50 = 3 nM T07173 C2A8TG 11978451 EC50 = 4 nM T07173 C0AVC3 12751666 EC50 = 667 nM T07173 CAW13S 16007060 IC50 < 1 nM T07173 CFPW41 16007116 Ki > 2500 nM T07173 C9JK2M 16059071 IC50 = 310 nM T07173 CW6UJ9 16059338 IC50 = 200 nM T07173 CH7MS6 16059729 IC50 = 170 nM T07173 CK0W2M 16097528 EC50 = 1 nM T07173 C20DST 16105503 IC50 > 1000 nM T07173 CCN62F 16105510 IC50 > 1000 nM T07173 CQG45C 16109001 IC50 = 8300 nM T07173 C1U8XW 16109036 IC50 = 18 nM T07173 CC5J0U 16112865 IC50 < 1 nM T07173 CGC34R 16118737 IC50 > 5000 nM T07173 C5VPH9 16129448 IC50 = 3510 nM T07173 CVZK29 16223008 IC50 = 350 nM T07173 CZ75LV 16259040 IC50 = 5000 nM T07173 CFC39H 16265338 IC50 = 775.2 nM T07173 C3XS1A 16267183 IC50 = 5000 nM T07173 CLZN74 16269984 IC50 = 2726.5 nM T07173 C9NV2A 16272977 IC50 = 517.3 nM T07173 C81LCV 16276659 IC50 = 12.1 nM T07173 C1ATH6 16322912 IC50 = 843.1 nM T07173 CY1E2N 16723801 IC50 > 100000 nM T07173 C2HVS1 16739794 IC50 = 2 nM T07173 C03EXR 16739855 IC50 = 2 nM T07173 CW64AB 16739883 IC50 < 1 nM T07173 CD7B6L 17561456 IC50 = 2449.6 nM T07173 CK7J6D 17756791 IC50 = 33000 nM T07173 CQ8UX6 18132565 IC50 = 13 nM T07173 C7HOI0 20907256 IC50 = 9085 nM T07173 CJPK63 20907257 IC50 > 9001 nM T07173 CJM18W 20966565 IC50 = 85 nM T07173 CE1TZ9 20971557 IC50 = 1287.4 nM T07173 CH4B5K 21081523 IC50 = 200 nM T07173 CT38MD 22170432 IC50 = 44 nM T07173 C6JV7W 23400934 IC50 > 7000 nM T07173 CD5S7O 23401001 IC50 = 8000 nM T07173 C8U6YG 24674418 IC50 = 5000 nM T07173 C7YG1N 24759534 IC50 = 310 nM T07173 CC69VF 24816435 IC50 = 7 nM T07173 CJ0CU5 24825841 IC50 = 8.24 nM T07173 C9B2TF 24880043 IC50 = 500 nM T07173 C5FD1A 24937369 IC50 > 500 nM T07173 C0KMW8 24937716 IC50 = 27 nM T07173 C5WG1H 24937847 IC50 = 21 nM T07173 CINE21 24948938 IC50 = 720 nM T07173 C0VMT7 24949091 IC50 = 360 nM T07173 C9PR3L 24949092 IC50 = 1900 nM T07173 CX56NK 24949093 IC50 = 13 nM T07173 C1WX3R 24949094 EC50 = 17 nM T07173 CYK54B 24949095 EC50 = 6 nM T07173 CN2IK6 24949096 EC50 = 81 nM T07173 CPM3Y9 24949243 EC50 = 3000 nM T07173 CDB6K7 24949244 EC50 = 2 nM T07173 CPA74B 24949245 EC50 = 9 nM T07173 C6ONY0 24949246 EC50 = 2 nM T07173 C5NVS6 24949247 IC50 = 750 nM T07173 C78RQK 24949248 IC50 = 1170 nM T07173 CBG64Q 24949398 IC50 = 100 nM T07173 C7IPT4 24949399 IC50 = 100 nM T07173 C0EH9D 24949400 IC50 = 650 nM T07173 C29VQI 24949401 IC50 = 120 nM T07173 CQ2TB6 24949402 EC50 = 20 nM T07173 C6DTP1 24949403 EC50 = 10 nM T07173 C3WL7Z 24949404 EC50 = 36 nM T07173 CUNL36 24949550 EC50 = 280 nM T07173 CI1GU4 24949551 EC50 = 1500 nM T07173 CJX82M 24949552 EC50 = 7 nM T07173 CGNY50 24949553 EC50 = 12 nM T07173 CEI2X1 24949554 EC50 = 3 nM T07173 C7Z6BJ 24949555 EC50 = 24 nM T07173 C0I3RP 24949705 EC50 = 60 nM T07173 CC6LM9 24949706 EC50 = 1 nM T07173 C8CO4B 24971342 IC50 = 270 nM T07173 C9OX4W 24971395 IC50 = 7 nM T07173 CGAR96 24971396 IC50 = 3 nM T07173 CKMV26 24971397 IC50 = 9 nM T07173 CMTY09 24971398 IC50 = 4 nM T07173 CERN39 24971399 IC50 = 52 nM T07173 C4WG5K 24971400 IC50 = 290 nM T07173 CTQR70 24971401 IC50 = 35 nM T07173 CZ46QO 24971402 IC50 = 110 nM T07173 C7VXE0 24971403 IC50 = 2600 nM T07173 C3KXQ5 24971404 IC50 > 5000 nM T07173 CMOZ41 24971405 IC50 > 5000 nM T07173 CQ58UR 24971406 IC50 = 610 nM T07173 CV5RY2 24971407 IC50 = 84 nM T07173 CP8J0I 24971408 IC50 = 10 nM T07173 CAJ9O3 24971409 IC50 = 118 nM T07173 CH5KQ3 24971410 IC50 = 1170 nM T07173 C8UE0S 24971411 IC50 = 111 nM T07173 C9F7BC 24971412 IC50 < 1 nM T07173 C4EG8R 24993189 IC50 > 10000 nM T07173 C3DI7Y 24995523 IC50 = 12 nM T07173 C6N7KR 25032700 IC50 = 0.6 nM T07173 CK4RG2 25167767 IC50 = 8 nM T07173 CQ04LW 25171665 IC50 = 1440 nM T07173 CU9KV5 25171666 IC50 = 670 nM T07173 CNG96H 25210579 IC50 > 10000 nM T07173 C2TXC6 25218656 IC50 > 500 nM T07173 CR5L9X 26012146 IC50 = 5000 nM T07173 C8P1KN 42105908 IC50 = 5000 nM T07173 CN8WB9 44189332 IC50 = 819 nM T07173 C3E7RP 44284203 IC50 = 61 nM T07173 C8FY7N 44284204 IC50 > 1000 nM T07173 CJH86A 44385063 IC50 = 61 nM T07173 CG46BQ 44386338 IC50 = 6 nM T07173 CA5M3C 44400503 IC50 = 4 nM T07173 C2U5IW 44412741 IC50 = 29 nM T07173 CZ4UV5 44446905 IC50 = 1900 nM T07173 C9GK5Z 44446906 IC50 = 1300 nM T07173 C2GQ8T 44446916 IC50 = 520 nM T07173 CML2R4 44446917 IC50 > 5000 nM T07173 CIQY85 44446918 IC50 > 5000 nM T07173 CUR09Q 44446919 IC50 = 790 nM T07173 CJ0HV9 44446920 IC50 > 5000 nM T07173 C9PUB4 44446921 IC50 = 2000 nM T07173 C2QIL9 44446922 IC50 = 1200 nM T07173 C32OCZ 44446923 IC50 = 760 nM T07173 CC1K4H 44446924 IC50 = 190 nM T07173 CP4O6S 44446925 IC50 = 320 nM T07173 C6MOS0 44446926 IC50 > 5000 nM T07173 CGVA97 44446927 IC50 = 2 nM T07173 CYB27I 44446928 IC50 = 67 nM T07173 C37RCI 44446929 IC50 = 10 nM T07173 C4Y8XV 44446930 IC50 = 31 nM T07173 CT91BO 44446931 IC50 = 60 nM T07173 CP9Z1O 44446932 IC50 = 720 nM T07173 CHO63P 44446933 IC50 = 1100 nM T07173 C8C1ZU 44446934 IC50 = 160 nM T07173 C98AGS 44446935 IC50 = 210 nM T07173 C3SQ8B 44446936 IC50 = 910 nM T07173 CB20MF 44446937 IC50 = 21 nM T07173 C39YBT 44446938 IC50 = 230 nM T07173 CZ6UA9 44446939 IC50 = 150 nM T07173 CWBV18 44446940 IC50 = 1 nM T07173 CPR51F 44446941 IC50 = 1 nM T07173 C85NEO 44448589 IC50 = 231 nM T07173 CG9YJ0 44448626 IC50 = 52 nM T07173 CKIA83 44448627 IC50 > 300 nM T07173 C5O9JU 44448658 IC50 > 300 nM T07173 C5W7LJ 44448659 IC50 = 43 nM T07173 CE5U6A 44448675 IC50 = 129 nM T07173 C7O6CF 44448676 IC50 = 49 nM T07173 CY1Q5B 44448696 IC50 = 33 nM T07173 C9W6ZO 44448697 IC50 = 14 nM T07173 CM4GV9 44448699 IC50 = 9 nM T07173 C92QJA 44448717 IC50 = 133 nM T07173 C76PSW 44518384 IC50 = 170 nM T07173 C6LP9V 44518674 IC50 = 75 nM T07173 CYH6P3 44520205 IC50 = 1870 nM T07173 C36KYB 44520611 IC50 = 68 nM T07173 CZH80Q 44520612 IC50 = 3130 nM T07173 CK49WN 45139234 IC50 = 910 nM T07173 CU3RF1 45139989 IC50 > 10000 nM T07173 CQGZ06 45139991 IC50 > 10000 nM T07173 C6OX0V 45375974 IC50 = 1480 nM T07173 CX0HO6 45486156 IC50 = 580 nM T07173 CY3HW5 46224684 IC50 > 10000 nM T07173 C7ON5A 46233287 IC50 > 10000 nM T07173 CM39AU 46275360 IC50 = 607 nM T07173 CU2X3I 46382263 IC50 = 1639.2 nM T07173 CBI7V6 46382265 IC50 = 216.8 nM T07173 CMP5T4 46382269 IC50 = 875.6 nM T07173 CRP7H0 46382271 IC50 = 44.7 nM T07173 CT5ZD0 46382272 IC50 = 126 nM T07173 COB29T 46382277 IC50 = 185.7 nM T07173 C7TY0M 46382278 IC50 = 20000 nM T07173 CUCX57 46382281 IC50 = 1107.1 nM T07173 CGR3T6 46382286 IC50 = 1843.7 nM T07173 CPZ81K 46382288 IC50 = 20000 nM T07173 CU9IK7 46382290 IC50 = 159.6 nM T07173 C61WCT 46382295 IC50 = 410.7 nM T07173 C4P1AT 46382302 IC50 = 6589.6 nM T07173 CMDC48 46382303 IC50 = 107.4 nM T07173 C2ZA3E 46382304 IC50 = 95 nM T07173 CN5R0P 46382305 IC50 = 227.9 nM T07173 CH53ZD 46382308 IC50 = 128.7 nM T07173 CT3UO5 46382309 IC50 = 65.9 nM T07173 C3R5DF 46382310 IC50 = 26.4 nM T07173 CVP36M 46382311 IC50 = 25.4 nM T07173 CEP0C1 46382312 IC50 = 271.2 nM T07173 CUG2W7 46382314 IC50 = 849 nM T07173 CDOR02 46382315 IC50 = 20000 nM T07173 CG6D4E 46382317 IC50 = 20000 nM T07173 C2L3WY 46382318 IC50 = 241.2 nM T07173 CPA41J 46382319 IC50 = 57.8 nM T07173 C54EDX 46382322 IC50 = 41.2 nM T07173 C9J1CQ 46382323 IC50 = 252.9 nM T07173 C37VDC 46382324 IC50 = 55 nM T07173 CG13SB 46382326 IC50 = 277.2 nM T07173 CD3QY0 46382327 IC50 = 24.5 nM T07173 C6ZNO1 46382331 IC50 = 163.4 nM T07173 CE6N3J 46382332 IC50 = 672.5 nM T07173 COD4I0 46382336 IC50 = 1820.8 nM T07173 CGD5Q0 46382338 IC50 = 5007.9 nM T07173 C40NSR 46382339 IC50 = 193.2 nM T07173 C8H2CR 46382341 IC50 = 167.1 nM T07173 C64RBV 46382343 IC50 = 142.3 nM T07173 C6NS1L 46382344 IC50 = 885.9 nM T07173 CP23VF 46382346 IC50 = 1457 nM T07173 CP9W3T 46382349 IC50 = 31.1 nM T07173 CZNH36 46382354 IC50 = 405.4 nM T07173 CYH93R 46382355 IC50 = 143.9 nM T07173 CV51XI 46382356 IC50 = 23.9 nM T07173 CVL8W3 46382358 IC50 = 5000 nM T07173 C7SKH2 46382366 IC50 = 164.8 nM T07173 CJD49N 46382375 IC50 = 327.1 nM T07173 CJ8E1N 46382394 IC50 = 444.4 nM T07173 CW4EI1 46390524 IC50 = 253.1 nM T07173 CQG51S 46390527 IC50 = 3744.9 nM T07173 CZ49OG 46390528 IC50 = 20000 nM T07173 CSJ20W 46390529 IC50 = 10000 nM T07173 CRAK47 46390532 IC50 = 20000 nM T07173 CQB16A 46872415 Ki > 4000 nM T07173 CLS29B 46872626 IC50 > 10000 nM T07173 C2O8RZ 46886323 IC50 > 1000 nM T07173 CCN08S 46934144 IC50 > 100000 nM T07173 CHSF07 49806372 IC50 = 261 nM T07173 CF91RS 49843531 IC50 > 10000 nM T07173 C8KT1S 50802118 IC50 = 41.5 nM T07173 C2X9OA 50802180 IC50 = 139.3 nM T07173 CF57GW 50802181 IC50 = 839.4 nM T07173 C1ED3N 50802184 IC50 = 5000 nM T07173 C6G1LV 50802187 IC50 = 20000 nM T07173 CC3YE6 50802196 IC50 = 5000 nM T07173 CBF28N 50802197 IC50 = 24.3 nM T07173 CK6G9M 50802198 IC50 = 38.2 nM T07173 CIC1B4 50802201 IC50 = 10.2 nM T07173 CWCP03 50802214 IC50 = 10000 nM T07173 CQP98F 50802215 IC50 = 247 nM T07173 CVT2O0 50802216 IC50 = 3030.3 nM T07173 C2G4HZ 50802217 IC50 = 5000 nM T07173 CB1AM0 50802226 IC50 = 32.4 nM T07173 CNRX75 50802227 IC50 = 5000 nM T07173 COJ6T7 50802228 IC50 = 20000 nM T07173 CH4K8I 50802229 IC50 = 5000 nM T07173 CST50B 50802232 IC50 = 10000 nM T07173 CI9H3K 50802245 IC50 = 20000 nM T07173 C1LHW9 50802246 IC50 = 7.7 nM T07173 C7IQV2 50802247 IC50 = 95 nM T07173 CY61RH 50802250 IC50 = 5000 nM T07173 CEA48B 50802259 IC50 = 51.1 nM T07173 CRT9S8 50802262 IC50 = 69.3 nM T07173 C23SQR 50802263 IC50 = 20000 nM T07173 C5IZR7 50802274 IC50 = 293.9 nM T07173 CVR8K4 50802276 IC50 = 2948.6 nM T07173 C4WMI1 50802277 IC50 = 21.1 nM T07173 CG52PC 50802293 IC50 = 79 nM T07173 CQ3R5U 50802295 IC50 = 19.3 nM T07173 CB3CE4 50802298 IC50 = 18.8 nM T07173 C3FYU7 50802299 IC50 = 59.1 nM T07173 C8A6MI 50802307 IC50 = 20000 nM T07173 C94SOF 50802309 IC50 = 11.5 nM T07173 C4Y6SN 50802310 IC50 = 6.8 nM T07173 CCKR79 50802312 IC50 = 5000 nM T07173 CFA79B 50802314 IC50 = 62.3 nM T07173 CB8PD0 50802328 IC50 = 5000 nM T07173 C17YAG 50802329 IC50 = 20.1 nM T07173 CSL61K 50802332 IC50 = 20000 nM T07173 CGBH51 50802345 IC50 = 2868.3 nM T07173 C13KBR 50802348 IC50 = 5000 nM T07173 C5SZE1 50802358 IC50 = 5000 nM T07173 C0F1XK 50802359 IC50 = 269 nM T07173 CE4HR6 50802360 IC50 = 242.9 nM T07173 CU5B4V 50802364 IC50 = 2.2 nM T07173 CV9PN1 50802374 IC50 = 1933 nM T07173 C17PKR 50802391 IC50 = 3935.7 nM T07173 CJ7G2O 50802392 IC50 = 4043.2 nM T07173 C5V3JC 50802393 IC50 = 5000 nM T07173 C8JKA9 50802404 IC50 = 9.1 nM T07173 C16UZW 50802409 IC50 = 60.3 nM T07173 C7KC5M 50802410 IC50 = 67.6 nM T07173 CX7BU6 50802411 IC50 = 5000 nM T07173 C5RI6H 50802419 IC50 = 5000 nM T07173 CR6GC8 50802420 IC50 = 5000 nM T07173 C6R1VG 50802424 IC50 = 5000 nM T07173 C6O9GD 50802433 IC50 = 41.2 nM T07173 C9UR2X 50825254 IC50 = 2711.6 nM T07173 C1UHX3 50825279 IC50 = 2585.2 nM T07173 C42SLF 50825281 IC50 = 5000 nM T07173 CGE97V 50825288 IC50 = 5000 nM T07173 CQ8D2T 50825304 IC50 = 5000 nM T07173 CWR12L 50825338 IC50 = 20000 nM T07173 CH6OS5 50825345 IC50 = 448.8 nM T07173 CVYM85 50825346 IC50 = 358.1 nM T07173 C2Y6QS 50938552 IC50 > 10000 nM T07173 C9NYP4 51036677 IC50 > 10000 nM T07173 C4WRY3 51037112 IC50 > 10000 nM T07173 CRI28Z 51037948 IC50 > 10000 nM T07173 CG5IK8 52936268 IC50 > 100000 nM T07173 C2CT5J 53236670 IC50 = 4500 nM T07173 C3M6LV 53236671 IC50 > 100000 nM T07173 CZ5L6F 53239373 IC50 > 100000 nM T07173 C2WFI8 53239374 IC50 > 100000 nM T07173 C0ZHF8 53239375 IC50 > 100000 nM T07173 CD1EQ3 53239587 IC50 = 12670 nM T07173 C0SWH5 53348216 IC50 > 40000 nM T07173 C8NA4L 53384644 IC50 = 29000 nM T07173 CE1ZK6 54759168 IC50 > 10000 nM T07173 CY3V6S 54764326 IC50 > 10000 nM T07173 CC7T2A 56674921 IC50 = 4700 nM T07173 C4Z0OC 56834890 IC50 = 200 nM T07173 C67TJQ 56834891 IC50 = 620 nM T07173 C1JLW8 57332840 IC50 = 3230 nM T07173 CD01JZ 57332841 IC50 = 5320 nM T07173 CCFK37 57332844 IC50 = 3720 nM T07173 CK1SR7 57332969 IC50 = 2480 nM T07173 C5TRE2 57332970 IC50 = 1450 nM T07173 C46TJK 57332974 IC50 = 7790 nM T07173 C09ZJY 57333095 IC50 = 9360 nM T07173 C8W6IG 57395117 IC50 > 30000 nM T07173 CU4FW8 57397383 IC50 = 7700 nM T07173 C59OYH 57398540 IC50 > 10000 nM T07173 C6U0SG 57629460 IC50 = 3 nM T07173 C1EVX0 58063117 IC50 = 3970 nM T07173 CSG5T1 58335664 IC50 = 5 nM T07173 CT3EW2 59292007 IC50 = 470 nM T07173 C7UZ4N 59397162 IC50 = 9 nM T07173 CXJ63M 59603829 IC50 = 540 nM T07173 CQEU96 59603842 IC50 = 50 nM T07173 CS19VO 59804294 IC50 = 9 nM T07173 CJ1BN7 59804319 IC50 = 7 nM T07173 CUQ6Y0 59804322 IC50 = 3 nM T07173 C8ZF3L 59804374 IC50 = 68 nM T07173 C6X2MP 60154732 IC50 = 47 nM T07173 CHOI42 60154733 IC50 = 18.6 nM T07173 CT29UY 60154734 IC50 = 64.7 nM T07173 CDT2N7 60154735 IC50 = 13.63 nM T07173 CJ94HK 60154736 IC50 = 8.36 nM T07173 CN2WV4 60154737 IC50 = 33.75 nM T07173 CVHT34 60154828 IC50 = 9.4 nM T07173 C63MQO 60154829 IC50 = 4.62 nM T07173 CG76XN 60154830 IC50 = 2.97 nM T07173 CQ4U2S 60154831 IC50 = 1.67 nM T07173 CIV8R9 60154832 IC50 = 5.41 nM T07173 CR07JV 60154833 IC50 = 110.3 nM T07173 CMDU45 60154921 IC50 = 3167 nM T07173 CFP86V 60155995 IC50 = 42.7 nM T07173 C8PQO7 60156000 IC50 = 69.6 nM T07173 CZVA50 60156001 IC50 = 31.4 nM T07173 CNT4Y7 60156097 IC50 = 26.47 nM T07173 C06MBL 60156098 IC50 = 22.7 nM T07173 CXC7S2 60156099 IC50 = 25.02 nM T07173 CW3CE6 60156100 IC50 = 33.2 nM T07173 C1YJG5 60156101 IC50 = 53.7 nM T07173 CCA2U4 60156102 IC50 = 22.2 nM T07173 CJ2EU8 60156103 IC50 = 88.6 nM T07173 CK6WO0 66552478 IC50 < 10000 nM T07173 C37NKO 67129970 IC50 > 10000 nM T07173 CK80LJ 67130050 IC50 > 10000 nM T07173 CV63UL 67240318 IC50 > 5000 nM T07173 CK31BI 67330085 IC50 = 2 nM T07173 C9ET6X 68310823 IC50 = 1.5 nM T07173 C0VJW8 68545858 IC50 = 50 nM T07173 C7GRV2 68755406 IC50 > 10000 nM T07173 C5DGR9 69036886 IC50 = 494 nM T07173 C3GTU1 69762142 IC50 > 10000 nM T07173 C7VJ6A 70647728 IC50 = 30 nM T07173 CT82EU 70681819 IC50 = 49 nM T07173 CX7Z2M 70688180 IC50 = 16 nM T07173 CT6CR8 70688181 IC50 = 27 nM T07173 CXZ40O 70696497 IC50 = 4 nM T07173 CGSX93 71212127 IC50 = 59 nM T07173 C7L0EM 71212130 IC50 = 118 nM T07173 C8UR7L 71212157 IC50 = 29 nM T07173 C76GHP 71212558 IC50 = 653 nM T07173 C1QY4Z 71212562 IC50 = 109 nM T07173 CFN2A6 71212571 IC50 = 12300 nM T07173 CV78TK 71454499 IC50 = 29 nM T07173 CKT60L 71455860 Ki > 2400 nM T07173 CCN01X 71547862 IC50 > 10000 nM T07173 C1NPL0 71552941 IC50 = 9790 nM T07173 CA4PS8 71552942 IC50 = 7710 nM T07173 CLCF69 72193625 EC50 = 6.5 nM T07173 C3IY6H 72204420 IC50 = 3 nM T07173 C8F2MQ 72206303 EC50 = 1005 nM T07173 CFI97M 73386687 IC50 = 997 nM T07173 C1V3NZ 73425588 IC50 = 1.67 nM T07173 CKAW05 73891123 IC50 < 100 nM T07173 CIQ5D8 74627727 IC50 = 47 nM T07173 CTXQ14 74627728 IC50 = 4233 nM T07173 CKU74R 74627729 IC50 = 2300 nM T07173 CPG3A5 86302574 IC50 > 30000 nM T07173 C1HW4B 89735655 IC50 = 2100 nM T07173 CK4EJ9 90014603 IC50 = 56 nM T07173 CQ2OB9 90292687 IC50 = 383 nM T07173 CHI39S 90292823 IC50 = 1550 nM T07173 CY0UC4 90645194 IC50 > 10000 nM T07173 CPH57U 90645509 IC50 = 11 nM T07173 CK6OT5 90645510 IC50 = 60 nM T07173 CN82QZ 90645511 IC50 = 7 nM T07173 CDMR53 90645512 IC50 > 100000 nM T07173 C10FPD 91666632 IC50 = 27 nM T07173 CI4N8P 91801232 IC50 = 0.3 nM T07173 CLZ74S 91826737 IC50 = 199 nM T07173 C0YVP7 91933872 IC50 = 0.16 nM T07173 C0Y8ZK 91933875 IC50 > 10 nM T07173 CC73YH 91933887 IC50 = 0.34 nM T07173 CJQ5N6 91936970 IC50 = 464000 nM T07173 CPGV73 101884319 IC50 = 22 nM T07173 CR17MP 101884320 IC50 = 3500 nM T07173 CA1TZ3 101884321 IC50 = 47 nM T07173 CG9KE7 101884322 IC50 = 39 nM T07173 C84MVD 101884325 IC50 = 24 nM T07173 C8OKH5 101884331 IC50 = 380 nM T07173 CS2JQ5 101884333 IC50 = 870 nM T07173 C3PAN1 117967296 IC50 = 99 nM T07173 CK9ZY1 117967567 IC50 = 4000 nM T07173 CX8W0E 117967965 IC50 = 28 nM T07173 CB3AU1 117967998 IC50 = 30 nM T07173 C5M6NG 117968174 IC50 = 4100 nM T07173 CT9F2D 117975098 IC50 = 82 nM T07173 CE86QC 118128728 IC50 = 2.7 nM T07173 C61WXP 118148480 IC50 = 6.1 nM T07173 C0TMZ8 118167692 IC50 = 1900 nM T07173 C68QVN 118167694 IC50 = 5400 nM T07173 CSM69G 118167758 IC50 = 720 nM T07173 C9EY8L 118167812 IC50 = 11 nM T07173 C4KC7H 118189484 IC50 = 3000 nM T07173 C5DYL3 118189493 IC50 = 74000 nM T07173 CLH8X7 118189551 IC50 = 7 nM T07173 CGN3D6 118392437 IC50 = 4 nM T07173 C1Z2BY 118393878 IC50 = 0.25 nM T07173 CF9U3Q 118394045 IC50 = 0.66 nM T07173 CBD7M6 118408591 IC50 = 1 nM T07173 CL0YO5 118443595 IC50 = 3.6 nM T07173 CF8C6D 118456250 IC50 = 1.99 nM T07173 CU3K0B 118456253 IC50 = 25 nM T07173 C2DS9I 118456276 IC50 = 16 nM T07173 C9ROH8 118497013 IC50 = 12 nM T07173 CQN74J 118497050 IC50 = 31 nM T07173 CP6N8V 118497084 IC50 = 4.7 nM T07173 CQ7A0F 118497113 IC50 = 34 nM T07173 CU9V4J 118497126 IC50 = 14 nM T07173 CL63AI 118497137 IC50 = 4 nM T07173 CN3AO5 118497153 IC50 = 14 nM T07173 C6BE3P 118497157 IC50 = 5 nM T07173 CBY47Z 118497161 IC50 = 74 nM T07173 CDG26L 118505207 IC50 = 1100 nM T07173 CC4ZE5 118505217 IC50 = 110 nM T07173 CP1IX9 118505219 IC50 > 50000 nM T07173 C4QE3G 118505223 IC50 = 41 nM T07173 C3QG0N 118505224 IC50 = 40 nM T07173 CP8B5K 118507002 IC50 = 23 nM T07173 C5FJ3B 118507004 IC50 = 120 nM T07173 CU02NF 118559124 IC50 = 32 nM T07173 C5K3SE 118590336 IC50 < 50 nM T07173 CTUK23 118590420 IC50 < 50 nM T07173 C1NYK8 118590483 IC50 < 50 nM T07173 CL74GH 118665602 IC50 = 28000 nM T07173 CP71CK 118665611 IC50 = 13000 nM T07173 CR3F5V 118665613 IC50 = 410000 nM T07173 C60TWO 118665627 IC50 = 7700 nM T07173 CY7T8F 118665628 IC50 = 61000 nM T07173 CY7BI2 118706214 IC50 > 10000 nM T07173 CQCX41 118737057 IC50 = 27 nM T07173 CPK47S 118868365 IC50 = 8.4 nM T07173 CN4X0C 121231414 IC50 = 68.4 nM T07173 CO19NG 121272655 IC50 = 215 nM T07173 CX5VD4 121272674 IC50 <= 0.7 nM T07173 CA6Z4R 121272745 IC50 = 70 nM T07173 CG7A1D 121277778 IC50 <= 0.9 nM T07173 CI21GB 121395217 IC50 < 10 nM T07173 C47KPV 121395220 IC50 < 10 nM T07173 C58SMZ 121395326 IC50 < 10 nM T07173 C08KEM 122179540 IC50 = 850 nM T07173 CQ43XF 122179541 IC50 = 740 nM T07173 C2TXZ9 122179542 IC50 = 170 nM T07173 CXS1Y6 122179543 IC50 = 76 nM T07173 CPF2L7 122179544 IC50 = 6 nM T07173 C3NJ6T 122179545 IC50 = 520 nM T07173 C3AJ4C 122179546 IC50 = 3 nM T07173 CG0RP7 122179547 IC50 = 1 nM T07173 C1A0SQ 122179548 IC50 = 3 nM T07173 C42GSX 122180520 Ki = 3600 nM T07173 C1HLE3 122183071 IC50 > 100000 nM T07173 CA21DQ 122183072 IC50 > 100000 nM T07173 CMT9I4 122183073 IC50 = 1600 nM T07173 CY0I8V 122183076 IC50 = 1100 nM T07173 CS53OG 122183080 IC50 = 420 nM T07173 CON46I 122183081 IC50 = 1700 nM T07173 CB0QF4 122183083 IC50 = 92 nM T07173 CTA36K 122183084 IC50 = 490 nM T07173 CE3D8I 122183086 IC50 = 530 nM T07173 CB2VY7 122183099 IC50 = 5 nM T07173 CZ1U4R 122183100 IC50 = 12 nM T07173 CQ89GW 122194424 IC50 = 88500 nM T07173 CB6MZ1 122194425 IC50 = 28900 nM T07173 CA2QJ8 122194426 IC50 = 117000 nM T07173 CKR76S 122194427 IC50 = 73300 nM T07173 CQU6T4 122194428 IC50 = 47200 nM T07173 CN3O6K 122194429 IC50 = 141000 nM T07173 CV79UD 122194430 IC50 = 6600 nM T07173 CE2ID0 122194431 IC50 = 14400 nM T07173 C4Y3PF 122194432 IC50 = 209000 nM T07173 CB48UY 122194433 IC50 = 10300 nM T07173 CD8UW2 122194434 IC50 = 16500 nM T07173 C9N7LP 122194435 IC50 = 16400 nM T07173 CS0N8C 122424459 IC50 < 100 nM T07173 C1XQE8 122424505 IC50 < 100 nM T07173 C31EKG 122424572 IC50 < 100 nM T07173 CC83HO 123131777 IC50 = 3300 nM T07173 CE51XL 126962607 IC50 = 30 nM T07173 C3HDB7 126962649 IC50 = 340 nM T07173 C54TNY 126962650 IC50 = 93 nM T07173 CZ3U6J 126962659 IC50 = 9.9 nM T07173 C3E7FZ 127028834 IC50 = 137 nM T07173 C0HN2Y 127030123 IC50 > 100000 nM T07173 C7S9GI 127030124 IC50 > 100000 nM T07173 CHGN68 127030424 IC50 = 3420 nM T07173 CRV62L 127030425 IC50 > 100000 nM T07173 CF7JT8 127030426 IC50 > 100000 nM T07173 C5YCU2 127030427 IC50 > 100000 nM T07173 C0GES2 127031075 IC50 > 100000 nM T07173 CFJ32Y 127031076 IC50 > 100000 nM T07173 CC8V4J 127031368 IC50 > 100000 nM T07173 C78GYH 127031383 IC50 > 100000 nM T07173 C5WA9Z 127031384 IC50 > 100000 nM T07173 CD7LN1 127031385 IC50 = 5810 nM T07173 CI0VX4 127031386 IC50 = 13740 nM T07173 CO89TC 127031387 IC50 = 1440 nM T07173 CAM4S5 127031675 IC50 = 6690 nM T07173 C4QD0M 127031676 IC50 = 9240 nM T07173 C0LTC3 127031677 IC50 > 100000 nM T07173 CO1G2K 127032542 IC50 > 100000 nM T07173 C12IOL 127033165 IC50 > 100000 nM T07173 C5RO0L 127033758 IC50 > 100000 nM T07173 CD04YX 127034308 IC50 > 100000 nM T07173 C0J6MA 129137802 IC50 < 10 nM T07173 CP1CK4 129137805 IC50 < 10 nM T07173 CCG89W 129148013 IC50 < 10 nM T07173 C0FM1R 130196825 IC50 = 110 nM T07173 C6IW3H 130200328 IC50 = 5.3 nM T07173 C35GFR 130200388 IC50 = 8.23 nM T07173 C57JRP 131839646 IC50 = 0.68 nM T07173 C12WSQ 132014694 IC50 = 2800 nM T07173 C4A1KN 132014906 IC50 = 10 nM T07173 CB9V6N 132015016 IC50 = 11 nM T07173 C93UNX 132041675 IC50 = 8.7 nM T07173 C6OXE3 132134663 IC50 >= 1000 nM T07173 CUO0C5 132156633 IC50 > 10000 nM T07173 CS9L3D 134147081 IC50 = 2 nM T07173 C90NWQ 134148467 IC50 = 48 nM T07173 C86MVT 134152794 IC50 = 20 nM T07173 C13BIY 134155803 IC50 = 13 nM T07173 C7HSO4 135407121 IC50 = 2545 nM T07173 C1QTS4 135459120 IC50 = 231.5 nM T07173 CV24UR 135873213 IC50 = 4000 nM T07173 CY2O5D 135883086 IC50 = 380 nM T07173 CHA4N2 136013680 IC50 > 10 nM T07173 CAW0E4 136065882 IC50 = 80630 nM T07173 C1YUD0 136219394 IC50 > 10 nM T07173 CIU8W3 136254389 IC50 > 10 nM T07173 CXC69T 137321158 IC50 = 26 nM T07173 CWC49K 137321210 IC50 > 1000 nM T07173 C3Z7BX 137355931 IC50 = 4.9 nM T07173 CO2P6J 137632400 IC50 = 9400 nM T07173 CW6G0M 137633567 IC50 = 14000 nM T07173 C7P8DL 137633612 IC50 > 81010 nM T07173 CI1E8V 137634241 IC50 = 5400 nM T07173 C6L3HN 137634634 IC50 = 31 nM T07173 C2YZA9 137634804 IC50 = 960 nM T07173 CS1J9F 137638576 IC50 = 2400 nM T07173 C1BC7X 137638843 IC50 > 81010 nM T07173 C0NKR4 137640958 IC50 = 49000 nM T07173 CB3R4E 137641283 IC50 > 81010 nM T07173 CPK38A 137642417 IC50 = 4394 nM T07173 CW3K1R 137642682 IC50 = 7310 nM T07173 CO0A5Z 137643316 IC50 = 99820 nM T07173 CHQ75A 137644894 IC50 = 74020 nM T07173 C0IS6J 137647123 IC50 = 64320 nM T07173 CAYP60 137647334 IC50 = 30870 nM T07173 C93MXU 137648253 IC50 = 662 nM T07173 CE0LZ1 137648904 IC50 = 36600 nM T07173 C8F4ZH 137649400 IC50 = 3388 nM T07173 CQ98LD 137650528 IC50 = 2552 nM T07173 C9YQS6 137652057 IC50 > 81010 nM T07173 C29VEU 137652242 IC50 = 11890 nM T07173 CH9BQ6 137653271 IC50 = 210 nM T07173 C48CER 137655170 IC50 = 22000 nM T07173 CD05EL 137655675 IC50 = 3944 nM T07173 CP87FM 137655709 IC50 = 880 nM T07173 C2A1BD 137656463 IC50 > 81010 nM T07173 CYG87D 137656818 IC50 > 81010 nM T07173 CC4GR1 137657302 IC50 = 218 nM T07173 CG5U3H 137657614 IC50 > 27000 nM T07173 CN3WV0 137657779 IC50 = 113 nM T07173 C7E9YA 137658125 IC50 = 12970 nM T07173 CIJZ70 137658859 IC50 = 47300 nM T07173 C8GQ4F 137659402 IC50 = 8829 nM T07173 CYVK51 137659623 IC50 = 1300 nM T07173 CIC3L2 137659789 IC50 = 961 nM T07173 CSWC68 137660376 IC50 > 81010 nM T07173 CJ0W9X 137660998 IC50 = 2114 nM T07173 CU9F5N 137661074 IC50 = 3163 nM T07173 CH12BE 138105933 IC50 = 730 nM T07173 C4Q9BD 138105934 IC50 = 1200 nM T07173 C8A4ZC 138105936 IC50 = 0.1 nM T07173 C0F9QE 138376543 IC50 = 26 nM T07173 C8WE0V 138454785 IC50 = 2600 nM T07173 CN0X5D 138454787 IC50 = 432 nM T07173 CP18OC 138455164 IC50 = 1.6 nM T07173 C4HUV3 138665084 IC50 = 23 nM T07173 CNRT47 139434032 EC50 = 550 nM T07173 CIN6L7 139434035 EC50 = 360 nM T07173 CTFE03 139434036 EC50 = 220 nM T07173 CX9H4W 139434047 EC50 = 780 nM T07173 CU10QZ 139434077 EC50 = 390 nM T07173 CLRW84 139434103 EC50 = 830 nM T07173 CB6F5R 139434105 EC50 = 1300 nM T07173 C7FBY1 139434107 EC50 = 340 nM T07173 C08MUD 139434127 EC50 = 220 nM T07173 C2MZ4L 139434198 EC50 = 500 nM T07173 CJIH42 139434200 EC50 = 230 nM T07173 C7W5MH 139434224 EC50 = 290 nM T07173 CXIT16 139434239 EC50 = 480 nM T07173 C2B8OV 139442846 EC50 = 180 nM T07173 C4ID6F 139442949 EC50 = 320 nM T07173 CX4E3H 142736778 IC50 = 3.81 nM T07173 CDA08X 145957845 IC50 = 8540 nM T07173 C6NT1H 145963881 IC50 = 1800 nM T07173 CAJQ14 145964002 IC50 = 20 nM T07173 CVF4M6 145965985 IC50 = 7.7 nM T07173 C1WA0P 145966817 IC50 = 40 nM T07173 C2P3YJ 145967230 IC50 = 8 nM T07173 CS9MZ3 145967758 IC50 = 1100 nM T07173 C5MHK6 145967970 IC50 = 2200 nM T07173 CK9C0H 145970062 IC50 = 23 nM T07173 C7PTX6 145973283 IC50 = 10 nM T07173 C6XV4Q 145974681 IC50 = 1 nM T07173 CI85EU 145998085 IC50 > 1000 nM T07173 CV8SQ4 155510804 IC50 < 10 nM T07173 C24NOX 155511218 IC50 = 18.1 nM T07173 CB5X7K 155511395 IC50 = 1700 nM T07173 CP6S7N 155511971 IC50 = 7.8 nM T07173 CDH4F9 155512717 IC50 = 1.1 nM T07173 CA10CQ 155512867 IC50 > 1000 nM T07173 C2MD1Q 155513187 IC50 > 10000 nM T07173 C5B2AX 155513312 IC50 = 7.34 nM T07173 CZMD64 155514443 IC50 > 1000 nM T07173 CB5T9G 155515436 IC50 = 326.3 nM T07173 CUK3M9 155516229 IC50 = 1.3 nM T07173 CX4L3U 155516368 IC50 = 110 nM T07173 CFV2I8 155516791 IC50 = 12.3 nM T07173 CUHZ87 155516883 IC50 > 1000 nM T07173 C6F5OW 155517096 IC50 = 1.04 nM T07173 COR4M0 155517181 IC50 = 264.4 nM T07173 CIU1T6 155518465 IC50 = 17.43 nM T07173 C86HPW 155518524 IC50 = 16000 nM T07173 CO63MP 155519543 IC50 = 2.65 nM T07173 C18ORE 155519760 IC50 < 10 nM T07173 C9TU2A 155520832 IC50 = 0.2 nM T07173 CSW1H4 155523508 IC50 = 48 nM T07173 CBG4P0 155524103 IC50 = 28.79 nM T07173 CV02BY 155526318 IC50 = 1.4 nM T07173 C9AG1S 155526843 IC50 = 2.7 nM T07173 CLJD37 155527082 IC50 = 0.89 nM T07173 CVQR59 155528115 IC50 = 15 nM T07173 CN6C2T 155528463 IC50 = 7.75 nM T07173 CQ40LX 155529074 IC50 = 253 nM T07173 C7QKS5 155529416 IC50 = 2.4 nM T07173 C2GQK7 155530525 IC50 = 175 nM T07173 C0HW7F 155530527 IC50 > 1000 nM T07173 CP5IW9 155530600 IC50 > 1000 nM T07173 C3MC2P 155532434 IC50 = 132.25 nM T07173 CNE6A3 155532801 IC50 = 39.78 nM T07173 C2KAU0 155533663 IC50 = 29.2 nM T07173 C75AKY 155533695 IC50 < 1 nM T07173 CQ6ZC2 155533969 IC50 = 95 nM T07173 C3PWI1 155534046 IC50 > 1000 nM T07173 C6K3BA 155535266 IC50 = 0.64 nM T07173 CTXK93 155535665 IC50 = 174 nM T07173 C14SEB 155535950 IC50 = 365.7 nM T07173 CV9D5J 155536164 IC50 = 186 nM T07173 CH6Z8W 155538581 IC50 = 1400 nM T07173 CN2Z1D 155539036 IC50 = 143.2 nM T07173 C3O6WX 155540330 IC50 > 1000 nM T07173 CLD3F7 155540396 IC50 = 120 nM T07173 C76NKG 155543431 IC50 > 1000 nM T07173 CEM59P 155543447 IC50 = 0.9 nM T07173 C38SPX 155545056 IC50 = 0.64 nM T07173 C12HEG 155545104 IC50 = 0.3 nM T07173 CRV40J 155546026 IC50 = 226.55 nM T07173 CPYV45 155546912 IC50 = 11.1 nM T07173 CBGI59 155547977 IC50 = 45 nM T07173 CU8C7A 155549730 IC50 = 1.02 nM T07173 C8AG4U 155550655 IC50 = 6.4 nM T07173 C2RQT8 155550913 IC50 < 1 nM T07173 CI2U8Q 155551163 IC50 = 0.59 nM T07173 C9MJL5 155551408 IC50 = 400 nM T07173 C6Z9DY 155551977 IC50 = 766.2 nM T07173 CM7Q3F 155556300 IC50 = 0.2 nM T07173 C25WDC 155556422 IC50 = 2.9 nM T07173 C9OLA3 155557330 IC50 = 0.2 nM T07173 C7RM5X 155560443 IC50 <= 0.5 nM T07173 CYD1C7 155560599 IC50 > 1000 nM T07173 C2DGR1 155561078 IC50 = 4.5 nM T07173 C40IYS 155562258 IC50 = 32.9 nM T07173 CN13EJ 155562386 IC50 = 7 nM T07173 CBG9Z1 155562952 IC50 = 398.3 nM T07173 C2ZI7W 155563158 IC50 = 3400 nM T07173 C0GF4I 155563533 IC50 < 100 nM T07173 C0WZ9S 155563842 IC50 > 1000 nM T07173 CWR4O5 155565233 IC50 = 3.56 nM T07173 CRFW02 155566430 IC50 = 41.61 nM T07173 C0V7SM 155567015 IC50 > 1000 nM T07173 C4QL2W 155567149 IC50 = 250 nM T07173 C8UDR0 155567423 IC50 < 100 nM T07173 CW18PH 155568478 IC50 = 264 nM T07173 CZSJ01 155568540 IC50 = 2.1 nM T07173 D00ERW 44444843 Ki > 2481 nM T07173 D00HVA 11624601 Ki > 2500 nM T07173 D02NNT 53232451 IC50 = 3 nM T07173 D02RWC 59397065 IC50 = 8 nM T07173 D02RWK 44400432 IC50 = 4 nM T07173 D03DYT 3035817 IC50 = 2.4 nM T07173 D03DZO 11715767 IC50 > 10000 nM T07173 D04RBG 3536 IC50 = 9 nM T07173 D07ADX 54764565 IC50 = 85 nM T07173 D07IHM 9823787 IC50 = 1055 nM T07173 D08HFG 24809764 IC50 > 10000 nM T07173 D09HVH 135566652 IC50 > 10 nM T07173 D09QBA 23378546 IC50 = 1270 nM T07173 D0D6MH 11617559 IC50 = 880 nM T07173 D0E7VO 59627005 IC50 = 1.4 nM T07173 D0J4YA 9943465 IC50 = 2 nM T07173 D0K5UF 72710568 IC50 = 17 nM T07173 D0L3JR 25212148 IC50 = 5 nM T07173 D0N4LR 53469448 IC50 = 1756 nM T07173 D0O8AR 16097523 Ki = 0.36 nM T07173 D0Q3NG 11715520 Ki > 2500 nM T07173 D0S7IE 11658882 Ki > 2500 nM T07173 D0T8NU 16757525 IC50 > 4000 nM T07173 D0US9O 45275255 IC50 = 35 nM T07173 D0Y4BL 11676971 IC50 = 15 nM T87661 CQTJ86 9547099 EC50 = 520 nM T87661 CIY57T 9547100 EC50 = 537.03 nM T87661 CE2FR8 52926276 EC50 = 1778.28 nM T87661 CK6IV9 52926277 EC50 = 770 nM T87661 CSV34F 52926278 EC50 = 288.4 nM T87661 C48ZQW 101780960 EC50 = 830 nM T87661 CVM0N2 122177490 EC50 = 1900 nM T87661 C0PF6Z 122177493 EC50 = 1995.26 nM T87661 CQ4H8Y 122177494 EC50 > 1000 nM T87661 CW9OA2 122177496 EC50 > 1000 nM T87661 CC43DK 122177497 EC50 > 1000 nM T87661 C2BWT6 122177498 EC50 > 1000 nM T87661 C4C1RL 122177499 EC50 > 1000 nM T87661 C5L3NY 122177503 EC50 > 1000 nM T87661 CEZN81 122177504 EC50 = 63 nM T87661 C6GHW5 122177506 EC50 = 1096.48 nM T87661 CAE7Y0 122177509 EC50 = 580 nM T87661 COD16Y 122177510 EC50 = 1047.13 nM T87661 CBI02Q 122177511 EC50 = 1548.82 nM T87661 CX27JM 122177512 EC50 > 1000 nM T87661 C2TQ8R 122177513 EC50 = 1348.96 nM T87661 CA0T9U 122177514 EC50 = 81.28 nM T87661 CZY0A1 122177515 EC50 = 489.78 nM T87661 CAZ90F 122177516 EC50 = 510 nM T87661 C4JP1B 122177517 EC50 = 43.65 nM T87661 C2GY9U 122177518 EC50 = 18 nM T87661 CX5EK3 122177519 EC50 = 75.86 nM T87661 CLD62P 122177520 EC50 = 33 nM T87661 CA8ZJ5 122177521 EC50 = 25 nM T87661 C67LAE 122177522 EC50 = 85.11 nM T87661 C30HEC 122177523 EC50 > 1000 nM T87661 CJ0RD5 122177524 EC50 > 1000 nM T87661 C6GI8E 122177525 EC50 > 1000 nM T87661 C0C5XU 122177526 EC50 > 1000 nM T87661 C74WRP 122177527 EC50 > 1000 nM T87661 C61RUZ 122177528 EC50 = 890 nM T87661 CRZ1V8 122177589 EC50 > 1000 nM T87661 C8XY1C 122177590 EC50 = 39.81 nM T87661 C6SGF5 122177591 EC50 = 720 nM T87661 CFLM72 122177592 EC50 = 30.9 nM T83982 CT0O5K 10634145 IC50 > 31600 nM T83982 C3Z5CV 46830074 IC50 > 200000 nM T83982 C8KCJ7 73659185 IC50 > 100000 nM T83982 CD96BW 73659186 IC50 > 100000 nM T83982 CEU7P1 86276129 IC50 > 100000 nM T83982 D0B0RZ 46174170 IC50 > 100000 nM T83982 D0I9UP 16065773 IC50 = 96 nM T84316 D0J0ZS 3446 IC50 = 27 nM T84316 CA6TL5 410547 IC50 = 220 nM T84316 CK8DN9 498058 IC50 = 960 nM T84316 C61FIK 715491 IC50 > 10000 nM T84316 CZ05PE 715493 IC50 = 180 nM T84316 C3G7VB 1234292 IC50 = 42 nM T84316 CFT04H 3056293 IC50 = 420 nM T84316 C32ABJ 9977389 IC50 = 107 nM T84316 CKDL43 9996195 IC50 = 170 nM T84316 CBZ5H9 10000286 IC50 = 737 nM T84316 C65JUQ 10000554 IC50 = 701 nM T84316 C5PYA6 10005269 IC50 = 1729 nM T84316 C1SX3M 10022126 IC50 = 86 nM T84316 C83ESN 10046621 IC50 = 153 nM T84316 C9PC4O 10051333 IC50 = 30 nM T84316 CPT29Q 10065679 IC50 = 171 nM T84316 CDK38E 10068070 IC50 = 528 nM T84316 C8NSO3 10069051 IC50 = 1597 nM T84316 C7Y3JG 10069052 IC50 = 4367 nM T84316 CLF9S1 10069697 IC50 = 440 nM T84316 C90HQI 10089184 IC50 = 185 nM T84316 CR8L0P 10089311 IC50 = 360 nM T84316 CJLV29 10249570 IC50 = 240 nM T84316 C52RPQ 10357989 IC50 = 250 nM T84316 CKO24Z 10380640 IC50 = 5180 nM T84316 CHWD90 10380703 IC50 = 40 nM T84316 CO0T6V 10406422 IC50 = 211 nM T84316 CZG3U4 10407905 IC50 = 335 nM T84316 CRB94W 10424606 IC50 = 1850 nM T84316 CM0Z8K 10428807 IC50 = 235 nM T84316 C5J2OV 10428813 IC50 = 9 nM T84316 CBIO09 10429369 IC50 = 75 nM T84316 C45CQE 10448940 IC50 = 170 nM T84316 C5OB1C 10450984 IC50 = 382 nM T84316 C35KYT 10452807 IC50 = 154 nM T84316 C4E7JS 10453204 IC50 = 577 nM T84316 CPG5V0 10455562 IC50 = 1263 nM T84316 CAF8E0 11152648 IC50 = 52 nM T84316 CPF64G 11156109 IC50 = 15 nM T84316 CGO4E9 11156110 IC50 = 198 nM T84316 C4EWI6 11166524 IC50 = 241 nM T84316 C45WVM 11190258 IC50 = 131 nM T84316 C3F6DV 11191376 IC50 = 29 nM T84316 CVZ60T 11213916 IC50 = 195 nM T84316 C3R2LI 11225909 IC50 = 183 nM T84316 C0JA1V 11235249 IC50 = 230 nM T84316 C29LOT 11237720 IC50 = 174 nM T84316 C2K5AJ 11245439 IC50 = 18 nM T84316 C0AUX3 11260400 IC50 = 10000 nM T84316 C9Z4GQ 11260702 IC50 = 829 nM T84316 CS67AJ 11271836 IC50 = 448 nM T84316 CBQK67 11271837 IC50 = 260 nM T84316 C3S7XG 11272151 IC50 = 116 nM T84316 C92CBZ 11305623 IC50 = 194 nM T84316 C9W8QX 11340838 IC50 = 1369 nM T84316 CT2V7A 11362278 IC50 = 145 nM T84316 CD3UC6 11363960 IC50 = 161 nM T84316 CP0M6U 11372899 IC50 = 1100 nM T84316 C9U7XS 11375307 IC50 = 700 nM T84316 CY7TH4 11398076 IC50 = 3163 nM T84316 CYC87R 11420562 IC50 = 291 nM T84316 CF4T2I 11450498 IC50 = 110 nM T84316 C1U7GA 11450937 IC50 = 38 nM T84316 CVO47R 11454689 IC50 = 145 nM T84316 CVXD25 11462217 IC50 = 270 nM T84316 COT41Y 11465156 IC50 = 342 nM T84316 CFLP46 11490010 IC50 = 28 nM T84316 CF70WY 11531673 IC50 = 30 nM T84316 C6DM5J 11596752 IC50 = 36 nM T84316 CWIN49 11725008 IC50 = 43 nM T84316 CSIB70 11775295 IC50 = 272 nM T84316 C1VD0L 11785247 IC50 = 630 nM T84316 CJH8M0 24788470 IC50 > 10000 nM T84316 CCK80G 40609282 IC50 = 11000 nM T84316 C2HM0W 44274811 IC50 = 2181 nM T84316 CY2ZK6 44299850 IC50 = 6000 nM T84316 CS01NJ 44300004 IC50 > 10000 nM T84316 CA3N0Y 44300010 IC50 = 160 nM T84316 CG8XC6 44300021 IC50 > 10000 nM T84316 C7J6AQ 44300028 IC50 = 5900 nM T84316 CDQH07 44300168 IC50 > 10000 nM T84316 C4KCY1 44300190 IC50 = 9900 nM T84316 CM54PQ 44300192 IC50 > 10000 nM T84316 CV6U5Z 44300214 IC50 = 5100 nM T84316 CI1Z7C 44300241 IC50 = 760 nM T84316 CE2Z0X 44407088 IC50 = 54 nM T84316 C1PDG9 44407089 IC50 = 161 nM T84316 CCH58F 44407095 IC50 = 84 nM T84316 CGJ6Z3 44407096 IC50 = 2926 nM T84316 C9KFM2 44407114 IC50 = 94 nM T84316 C1BH7N 44407115 IC50 = 37 nM T84316 COQ5I9 44407117 IC50 = 65 nM T84316 CB1KU4 44407120 IC50 = 144 nM T84316 CB82IJ 44407121 IC50 = 84 nM T84316 CML9T2 44407131 IC50 > 3000 nM T84316 CRZ92G 44407141 IC50 = 296 nM T84316 CK81AL 44407154 IC50 = 32 nM T84316 C0F9MZ 44407158 IC50 = 84 nM T84316 CGR5P1 44407159 IC50 = 18 nM T84316 C7HA5K 44407173 IC50 = 702 nM T84316 C6SQE1 44407174 IC50 = 76 nM T84316 CD0TN9 44407178 IC50 = 63 nM T84316 C3O6AD 44407179 IC50 = 153 nM T84316 C3U8DH 44407183 IC50 = 179 nM T84316 C70FBZ 44407184 IC50 = 180 nM T84316 C6RS4M 44407192 IC50 = 70 nM T84316 C0P8QN 44407195 IC50 = 67 nM T84316 CI5QZ2 44407196 IC50 = 61 nM T84316 CV2AG5 44407201 IC50 = 221 nM T84316 CIOA21 44407208 IC50 = 370 nM T84316 CPOD40 44407209 IC50 = 702 nM T84316 C7VLW4 44407216 IC50 = 1692 nM T84316 C61PQW 44407222 IC50 = 239 nM T84316 CMS4W2 44407242 IC50 = 199 nM T84316 CU38MP 44407245 IC50 = 207 nM T84316 CBMT74 44407252 IC50 = 50 nM T84316 CRG3Y5 44407253 IC50 = 84 nM T84316 CTH48Q 44407255 IC50 = 69 nM T84316 CJ41NQ 44407256 IC50 = 119 nM T84316 C0J3UB 44407259 IC50 = 64 nM T84316 C9D3YX 44407268 IC50 = 346 nM T84316 C64IKW 44407285 IC50 = 68 nM T84316 CDHB39 44407304 IC50 > 3000 nM T84316 C4SJ9F 44459324 IC50 = 597 nM T84316 CV89DA 44459491 IC50 > 10000 nM T84316 CIX47S 44459729 IC50 = 263 nM T84316 CD75KV 44459734 IC50 = 148 nM T84316 CY93SX 44459781 IC50 > 10000 nM T84316 CB2PZ0 44459869 IC50 > 10000 nM T84316 CB53AF 44460966 IC50 = 10000 nM T84316 CZN6H5 44461091 IC50 = 220 nM T84316 CG7UO8 44461104 IC50 = 36 nM T84316 CWI61J 44461267 IC50 = 72 nM T84316 CBK4Z8 44461344 IC50 = 229 nM T84316 CN4P9E 44461345 IC50 = 10000 nM T84316 CA2JU7 46911115 IC50 = 8 nM T84316 C73VYX 46911116 IC50 = 8 nM T84316 CVD43F 56659471 IC50 = 6 nM T84316 C8SR2X 56659475 IC50 = 2 nM T84316 CNM68T 56662903 IC50 = 169 nM T84316 CP2LW0 56662936 IC50 = 32 nM T84316 CX9FB0 56662937 IC50 = 200 nM T84316 C8PQ0U 56666408 IC50 = 3 nM T84316 C7BQD3 56669824 IC50 = 5 nM T84316 CHAK86 56669827 IC50 = 213 nM T84316 CU0KW5 56673309 IC50 = 32 nM T84316 CDX09S 56673310 IC50 = 5 nM T84316 CK8U1S 56673311 IC50 = 79 nM T84316 C0OYQ1 56676613 IC50 = 58 nM T84316 C04IVB 56676641 IC50 = 32 nM T84316 CW37HG 56676642 IC50 = 25 nM T84316 CLF76V 56676643 IC50 = 3 nM T84316 C4QCS7 56676649 IC50 = 1 nM T84316 CZ98WA 56676650 IC50 = 22 nM T84316 C8QO3N 56679972 IC50 = 20 nM T84316 C4CY2J 56679973 IC50 = 126 nM T84316 C7TR6Q 56679975 IC50 = 22 nM T84316 CMWY31 56683305 IC50 = 2 nM T84316 CY5S9E 56683306 IC50 = 25 nM T84316 C3J2FI 56683309 IC50 = 7 nM T84316 D0VQ4G 44300061 IC50 = 13000 nM T03755 D00PBX 49846579 Ki = 245 nM T03755 D02OZK 11404337 Ki = 1000 nM T03755 D06ETI 24978538 IC50 = 70 nM T03755 D0Z0HH 3503 Ki = 17700 nM T03755 D0L8WH 11228183 Ki <= 1 nM T03755 C5KW4H 72311 Ki = 106000 nM T03755 CBXG18 245869 Ki = 127000 nM T03755 CRV86S 1555114 Ki = 243000 nM T03755 CJ5TR3 1576659 Ki = 21500 nM T03755 CGAM30 1582605 Ki = 37530 nM T03755 CRP38E 4369509 IC50 > 25000 nM T03755 CR2V0Y 6090108 Ki = 124000 nM T03755 CJU75C 7655492 Ki = 31200 nM T03755 CQSY92 11546381 IC50 = 8090 nM T03755 C34ZAH 16072153 Ki = 54200 nM T03755 CHP79I 16109159 Ki = 49 nM T03755 C5NI1B 24798804 IC50 = 440 nM T03755 CU34VF 25232834 IC50 = 5000 nM T03755 C68YHX 26378673 Ki = 610000 nM T03755 C6GOQ2 27433194 Ki = 88000 nM T03755 CP7O6U 44286285 Ki = 59320 nM T03755 CB8P9H 44409349 IC50 = 26850 nM T03755 CB7V0S 44409350 IC50 = 13990 nM T03755 C5N2AO 44429172 Ki = 41100 nM T03755 CC5MY2 44429173 Ki = 24100 nM T03755 CO35QT 44429175 Ki = 58300 nM T03755 CR40TC 44429176 Ki = 61900 nM T03755 CDK47L 44429177 Ki = 6980 nM T03755 C4UFY2 44429178 Ki > 1000000 nM T03755 CMT5V4 44429179 Ki = 146000 nM T03755 C2XAH8 44429180 Ki = 56800 nM T03755 CRV49G 44429181 Ki = 116000 nM T03755 CG35DU 44456125 Ki = 116000 nM T03755 CLF8A1 44456175 Ki = 88300 nM T03755 C59ZEM 44456176 Ki = 39200 nM T03755 CAZ5T0 44456210 Ki = 101000 nM T03755 CV43WR 44456211 Ki = 99000 nM T03755 C85FLZ 44456249 Ki = 13700 nM T03755 C4W6OL 44456329 Ki = 2200 nM T03755 C5MP1Y 44456362 Ki = 2300 nM T03755 CHKW90 44456365 Ki = 1300 nM T03755 CH3KZ7 44567885 Ki = 12950 nM T03755 CLR6W0 44567922 Ki = 10800 nM T03755 COL2S9 44567923 Ki = 9430 nM T03755 CH2E4R 44609307 Ki = 1920 nM T03755 C2ZT6I 51354614 IC50 > 1000 nM T03755 C73DOP 51354615 IC50 = 245 nM T03755 CNA1W2 51354616 IC50 > 1000 nM T03755 C4Q3YN 51354902 IC50 = 540 nM T03755 CON3Q1 51354903 IC50 > 1000 nM T03755 C52OHD 51354904 IC50 = 275 nM T03755 CM3CU0 51355193 IC50 > 1000 nM T03755 CUK97J 57392876 Ki = 170 nM T03755 C1MQF6 57392877 Ki = 59 nM T03755 C38WES 57392878 Ki = 21 nM T03755 C5XZ9E 57396359 Ki = 63 nM T03755 CD0YR1 57403327 Ki = 55 nM T03755 CBLR64 59447577 Ki = 19 nM T03755 CP3Y2O 71548702 Ki = 1360 nM T03755 CS02CG 71549001 Ki = 2190 nM T03755 C37AJW 71549412 Ki = 4410 nM T03755 C16WOR 72715983 IC50 > 25000 nM T03755 C7O1BG 73347486 IC50 = 5000 nM T03755 CVC6Z1 73349009 IC50 > 10000 nM T03755 C6KWN5 73349012 IC50 > 10000 nM T03755 C6ZGJ8 73353547 IC50 > 10000 nM T03755 C3C7QO 86765310 Ki = 1580 nM T03755 C5W2EA 118734957 Ki > 660 nM T03755 CB37YD 155518816 IC50 = 59100 nM T03755 CNAR96 155536134 IC50 = 4010 nM T03755 CK7UQ4 155537237 IC50 = 4370 nM T03755 C6TQ4X 155545656 IC50 = 14500 nM T03755 CUX0F2 155558443 IC50 = 21000 nM T03755 C5Y0QF 155565915 IC50 = 12500 nM T03755 C8CL3Z 155569283 IC50 = 1000 nM T03755 D05RDP 992586 Ki = 8190 nM T03755 D0V7PX 454878 Ki = 2100 nM T36147 CRTI09 3281693 IC50 = 7000 nM T36147 CMZ3Y7 3281697 IC50 = 10000 nM T36147 C2FV5I 3676137 IC50 = 10000 nM T36147 CAIN92 3676139 IC50 = 5000 nM T36147 C47RMQ 4738040 Ki = 20.8 nM T36147 C4IC9P 5052527 IC50 > 100000 nM T36147 CX7PR4 14449988 Ki = 0.00329 nM T36147 CE2S3V 14449989 Ki = 0.00227 nM T36147 CH09BS 14449992 Ki = 0.00327 nM T36147 CO18RX 15994611 IC50 = 51000 nM T36147 CN73KG 15995634 IC50 = 20000 nM T36147 C13GDN 15995636 IC50 = 36000 nM T36147 CKBP83 16002078 IC50 = 24000 nM T36147 CTW8E4 22421659 IC50 = 21000 nM T36147 C8FVN2 44364233 IC50 > 30000 nM T36147 CZ04YN 44364234 IC50 > 30000 nM T36147 C3O6CP 44364235 IC50 > 30000 nM T36147 C26UCS 44364243 IC50 = 900 nM T36147 C6U1OH 44364244 IC50 = 700 nM T36147 C4U5PA 44364245 IC50 = 80 nM T36147 C61JHV 44364339 IC50 = 50 nM T36147 CWKU04 44364360 IC50 = 60 nM T36147 CA3BD4 44364376 IC50 = 200 nM T36147 CU6L0D 44364420 IC50 = 40 nM T36147 CXR49U 44364421 IC50 > 30000 nM T36147 CU4AE5 44436348 Ki = 500000 nM T36147 C5WE1G 46504414 IC50 = 18000 nM T36147 C35BOE 56589587 Ki = 20000 nM T36147 CIUK84 68295193 IC50 > 100000 nM T36147 C8MDV0 71450599 IC50 = 67000 nM T36147 C4TS3K 71450625 Ki = 0.00217 nM T36147 CT18ZB 71450627 Ki = 0.00636 nM T36147 C9H5UW 71450628 Ki = 0.000589 nM T36147 CE2GY7 71450629 Ki = 0.00653 nM T36147 CO96LQ 71450630 Ki = 0.0044 nM T36147 CLOH40 71452463 Ki = 0.000288 nM T36147 CO0CD2 71452464 Ki = 0.00302 nM T36147 CT8XK3 71454219 Ki = 0.00759 nM T36147 C8JB7E 71455954 IC50 = 30000 nM T36147 CLEN68 71455977 Ki = 0.001 nM T36147 CY36VC 71455978 Ki = 0.011 nM T36147 CIT25C 71457753 IC50 = 146000 nM T36147 C1H8RS 71457776 Ki = 0.0017 nM T36147 CW9IG1 71457777 Ki = 0.0333 nM T36147 CV7EO8 71457778 Ki = 0.012 nM T36147 CLAP24 71459674 IC50 = 30000 nM T36147 C0L4GC 71459695 Ki = 0.00153 nM T36147 CU79DN 71459696 Ki = 0.00445 nM T36147 CTC3X4 71463143 Ki = 0.00411 nM T36147 C2LX6O 92208905 IC50 = 10000 nM T36147 CMSX05 136216669 Ki = 1.33 nM T85915 CPO5K4 23633257 EC50 = 560 nM T85915 CK6N2D 24894761 EC50 = 750 nM T85915 CZBX15 24894990 EC50 = 800 nM T85915 C5CMV4 44560969 EC50 = 1190 nM T85915 CL2BP0 117947705 IC50 = 7 nM T00577 D09FAZ 9444 IC50 = 300 nM T00577 D0U5SI 4913 IC50 > 500000 nM T00577 D0X5XU 451668 IC50 = 30 nM T00577 D0L4FS 5280961 IC50 = 30000 nM T00577 D0U2BH 65064 IC50 = 500 nM T00577 D02VTV 117968550 EC50 = 100000 nM T00577 D03LZO 117967861 EC50 = 46000 nM T00577 C5IO2D 171251 IC50 > 45000 nM T00577 CKS4U8 188380 IC50 = 302000 nM T00577 CJH6D9 327606 IC50 = 100000 nM T00577 CA6J0D 445762 IC50 = 18000 nM T00577 C3KVN2 702558 IC50 = 390000 nM T00577 CQEF34 1002773 IC50 > 100000 nM T00577 CJ4ID2 3718032 IC50 = 12000 nM T00577 CG0D6N 10451940 IC50 > 100000 nM T00577 CZC4W3 11576752 IC50 = 27000 nM T00577 CIC81U 21120307 IC50 = 45000 nM T00577 CDMU19 24828467 IC50 = 150000 nM T00577 C85NAQ 24858111 IC50 = 850 nM T00577 C2ENB5 24947577 IC50 = 18000 nM T00577 C6D0LY 30118838 IC50 = 20000 nM T00577 CW7Z9B 45267108 IC50 = 6000 nM T00577 CBYR03 45267109 IC50 = 31000 nM T00577 C4YJQ9 45267958 IC50 > 10000 nM T00577 CYBW25 45267964 IC50 = 216000 nM T00577 CR4BF6 45267973 IC50 = 7400 nM T00577 CL0JD3 45267974 IC50 = 820 nM T00577 C70YFN 45267975 IC50 = 36000 nM T00577 CGYV47 45267981 IC50 = 22000 nM T00577 CP1OF8 45268848 IC50 = 75000 nM T00577 C7T2ZU 45268859 IC50 = 5000 nM T00577 CT84RL 45269774 IC50 > 100000 nM T00577 CX6H5T 45270517 IC50 = 8000 nM T00577 CE7K6J 45270523 IC50 = 154000 nM T00577 CR5B0C 45270527 IC50 = 5400 nM T00577 C54CSO 45270528 IC50 = 3700 nM T00577 C90XJH 45270533 IC50 = 6700 nM T00577 C6YIP2 45270600 IC50 = 8000 nM T00577 CK8BR2 45271342 IC50 = 44000 nM T00577 CCV8K1 45271353 IC50 = 44000 nM T00577 CHE5I6 45271416 IC50 > 100000 nM T00577 CQP6C4 45271423 IC50 = 300000 nM T00577 C87VSU 45272236 IC50 = 2500 nM T00577 CWD34S 45272237 IC50 = 4500 nM T00577 C2PUO3 45272238 IC50 = 4800 nM T00577 CL19VE 45272250 IC50 = 15000 nM T00577 CZJ86D 45272318 IC50 > 100000 nM T00577 CD47UG 45272319 IC50 = 4000 nM T00577 C83FZD 45273085 IC50 = 45000 nM T00577 C2YXN3 45273086 IC50 = 2900 nM T00577 C5MO1Y 45273087 IC50 = 21000 nM T00577 CDJE90 45273088 IC50 > 100000 nM T00577 CRE09G 45273096 IC50 = 19000 nM T00577 CWO9X2 45273097 IC50 = 94000 nM T00577 CIX92D 45273102 IC50 = 61000 nM T00577 C7E9SW 45273103 IC50 = 2500 nM T00577 CN96GS 45273186 IC50 = 1100 nM T00577 C03YWX 49786972 Ki > 50000 nM T00577 CPL71I 54596764 IC50 = 121000 nM T00577 CFY18X 56643471 IC50 = 150000 nM T00577 C32POU 56648592 IC50 = 270000 nM T00577 C0IPV6 56648595 IC50 = 1600000 nM T00577 C2AP8B 56648690 IC50 = 570000 nM T00577 CXBY54 56648693 IC50 = 310000 nM T00577 CQ34RM 56648770 IC50 = 1130000 nM T00577 C0XFZ5 56935564 IC50 = 4000 nM T00577 CJBY70 56951879 IC50 = 2.9 nM T00577 CB49HN 59457966 IC50 = 173000 nM T00577 C7M0FJ 59457983 IC50 = 370 nM T00577 CER5F1 67466175 IC50 > 100000 nM T00577 CO3F1Q 70686507 IC50 = 22000 nM T00577 C62WVR 70695988 IC50 = 132000 nM T00577 C9NV1Z 76310239 IC50 = 98000 nM T00577 CJ8H5F 76310241 IC50 = 40000 nM T00577 C52YJT 76310995 IC50 = 4110 nM T00577 CD1M0Q 76313934 IC50 = 20000 nM T00577 CNQ86R 76314627 IC50 = 174000 nM T00577 CAKL96 76314628 IC50 = 68000 nM T00577 CYB1U4 76318201 IC50 = 9000 nM T00577 C18MDV 76321200 IC50 = 80000 nM T00577 CZ09ML 76321898 IC50 = 35000 nM T00577 CF3KG5 76325534 IC50 = 38600 nM T00577 C4OYL7 76325535 IC50 = 27900 nM T00577 C08QPM 76328372 IC50 = 73000 nM T00577 CFX2B7 76328373 IC50 = 230000 nM T00577 CA54DX 76332046 IC50 = 128000 nM T00577 C84NAS 76332047 IC50 = 50000 nM T00577 CY05NB 76332742 IC50 = 12300 nM T00577 CDL08Z 76336365 IC50 = 650 nM T00577 C4XJ5N 78357767 IC50 > 100000 nM T00577 C01DAP 86288828 IC50 = 179000 nM T00577 CVM64R 117967504 EC50 = 30000 nM T00577 CJY5W0 117967660 EC50 = 73000 nM T00577 CM5N2A 117967691 EC50 = 27000 nM T00577 C2G4ND 117967705 EC50 = 26000 nM T00577 CY1V9T 117976066 EC50 = 32000 nM T00577 CY2R4J 117976176 EC50 = 20000 nM T00577 CSTY10 118607373 IC50 = 73 nM T00577 C9BI8F 118607414 IC50 = 619 nM T00577 CSW92P 118607432 IC50 = 382 nM T00577 CO1D7I 118607435 IC50 = 4420 nM T00577 C6PZ1X 118607459 IC50 = 750 nM T00577 CBA79J 118607465 IC50 = 645 nM T00577 CLS25W 118607471 IC50 = 494 nM T00577 C1K0VJ 118607474 IC50 = 1370 nM T00577 C8XMV5 118607488 IC50 = 497 nM T00577 CY1X2K 118613614 IC50 = 950 nM T00577 CT6OD8 118613615 IC50 = 1070 nM T00577 COPW27 118613616 IC50 > 10000 nM T00577 CJW05H 118613617 IC50 = 978 nM T00577 C7X2AQ 118613624 IC50 = 413 nM T00577 CE69HN 118613626 IC50 = 297 nM T00577 CDK3F2 118613628 IC50 = 1080 nM T00577 C5AF9V 118613631 IC50 = 1050 nM T00577 CG39ZR 118613632 IC50 = 582 nM T00577 CUDE80 118613633 IC50 = 969 nM T00577 CLIZ07 118613634 IC50 = 230 nM T00577 CG6E0J 118613636 IC50 = 1050 nM T00577 C07LSQ 118613637 IC50 = 1410 nM T00577 CB0K3S 118613639 IC50 = 232 nM T00577 C7SIL0 118613641 IC50 = 1250 nM T00577 CQD69N 118613646 IC50 = 234 nM T00577 CQNA84 118613647 IC50 = 201 nM T00577 CBC0Q9 118613651 IC50 = 290 nM T00577 C2EQ9X 118613653 IC50 = 140 nM T00577 C1X8GW 118613658 IC50 = 123 nM T00577 C0JVC9 118613660 IC50 = 957 nM T00577 CI70WP 118613691 IC50 = 316.23 nM T00577 CQ5T3E 118613693 IC50 > 10000 nM T00577 CFGK68 118613694 IC50 = 618 nM T00577 C1LOF4 118613696 IC50 = 759 nM T00577 CAY5Q6 118613697 IC50 = 1600 nM T00577 CG7D9I 118613701 IC50 = 945 nM T00577 C3ZJO5 118613702 IC50 = 2290 nM T00577 COJB60 118613705 IC50 = 929 nM T00577 CX8J7D 118613718 IC50 = 1270 nM T00577 CKI70Y 118613722 IC50 = 624 nM T00577 CJY8E1 118613723 IC50 = 781 nM T00577 CPW12K 118613724 IC50 = 1030 nM T00577 C3QX6D 118613726 IC50 = 137 nM T00577 CKO15P 118613728 IC50 = 1790 nM T00577 CW1D6K 118613729 IC50 = 32 nM T00577 CGQ82T 118732749 IC50 = 19000 nM T00577 CV0FW8 121225442 IC50 = 150 nM T00577 C6G0CZ 122580323 EC50 > 100000 nM T00577 CJI14M 129072680 IC50 = 21 nM T00577 CU3FP1 129072681 IC50 = 83 nM T00577 C0ES4L 129072695 IC50 = 588 nM T00577 COL81P 129085358 IC50 = 40 nM T00577 CUZ6K0 129085359 IC50 = 2080 nM T00577 CI1H4A 129085361 IC50 = 298 nM T00577 C2B5VP 129085364 IC50 = 274 nM T00577 CJ18GA 129085365 IC50 = 247 nM T00577 CUO5E6 129085366 IC50 = 425 nM T00577 CVPH43 129085367 IC50 = 212 nM T00577 CKS08I 129085368 IC50 = 446 nM T00577 CNO1K2 129085369 IC50 = 414 nM T00577 CIST32 129085377 IC50 = 200 nM T00577 CL9KB8 129246684 IC50 = 1870 nM T00577 C6ZYB8 129270457 IC50 = 1320 nM T00577 CL0WR7 134386479 EC50 > 100000 nM T00577 C5H9YP 135398693 IC50 > 1000000 nM T00577 C6GC0O 137028680 EC50 > 100000 nM T00577 C4S1ZI 137333995 IC50 = 3100 nM T00577 CWMH49 137638632 EC50 = 16000 nM T00577 C05DFP 137653852 EC50 = 24000 nM T00577 C95RGF 145950703 IC50 = 231 nM T00577 C0XBU5 145951018 IC50 = 284 nM T00577 CIKY95 145954902 IC50 = 2250 nM T00577 C5NS1C 145963999 IC50 = 475 nM T00577 CMX3R9 145964677 IC50 = 722 nM T00577 C7XF6P 145965645 IC50 = 501 nM T00577 CW2ZV7 145967174 IC50 = 80 nM T00577 C39OCT 145967367 IC50 = 494 nM T00577 C3JO8Q 145971403 IC50 = 187 nM T00577 COJG25 145974212 IC50 = 261 nM T00577 CKVI47 145974419 IC50 = 83 nM T00577 CW1LX9 145975217 IC50 = 235 nM T00577 CIP42V 145976082 IC50 = 211 nM T00577 C8MFK6 145977537 IC50 = 205 nM T00577 C5I0ZL 145977690 IC50 = 833 nM T00577 CU2A1M 145978072 IC50 = 234 nM T00577 C3MF6X 145978745 IC50 = 250 nM T00577 CUVO30 155515610 EC50 > 100000 nM T00577 CX5G9E 155528619 EC50 > 100000 nM T00577 CS3PF1 155533577 EC50 > 100000 nM T00577 CRH9J5 155534178 EC50 > 100000 nM T00577 CAE51Q 155534378 EC50 > 100000 nM T00577 C29RHJ 155544579 EC50 > 100000 nM T00577 CIN57Q 155556138 IC50 = 14000 nM T00577 CB8SD4 155557649 EC50 > 100000 nM T00577 C0BU1J 155560963 EC50 > 100000 nM T00577 D02TVQ 71268957 IC50 > 100000 nM T00577 D06PPL 25150857 IC50 > 10000 nM T00577 D07VWC 344265 IC50 = 50000 nM T00577 D08TGQ 124349 IC50 = 1500 nM T00577 D09CLP 439155 IC50 = 4000 nM T00577 D0A2ZH 266989 IC50 = 212000 nM T00577 D0BI4T 53315878 IC50 > 50000 nM T00577 D0GK7A 46224516 IC50 = 1287 nM T00577 D0I2RW 8342 IC50 = 1600 nM T00577 D0J5VK 67145 IC50 = 47000 nM T00577 D0L0DC 53339032 Ki = 950 nM T00577 D0S9SJ 56962337 IC50 = 0.3 nM T90782 D01BYB 5957 EC50 > 100000 nM T90782 D07QQP 10219163 EC50 > 1000 nM T90782 D0H2UB 5361 IC50 = 27000 nM T90782 D0S6AE 148197 EC50 = 1160 nM T90782 D0Z7FU 6133 EC50 = 424 nM T90782 C9K3IP 78253 IC50 > 10000 nM T90782 CS2M9I 148196 EC50 = 2000 nM T90782 C6VB7R 150973 EC50 > 1000 nM T90782 CM6QD5 189010 EC50 = 7560 nM T90782 CO6A2E 451388 EC50 = 140 nM T90782 C7NR6U 3081495 EC50 > 100000 nM T90782 C6P7VU 5311303 EC50 > 100000 nM T90782 CRK8Q6 9853990 EC50 = 2030 nM T90782 CVZX40 9875011 EC50 = 270 nM T90782 CR4UQ9 9875516 EC50 = 950 nM T90782 C2F7DR 10098947 EC50 = 9750 nM T90782 CN3Q7U 10207117 EC50 = 333 nM T90782 CO0L9C 10234467 EC50 > 10000 nM T90782 CF08GK 10432343 EC50 = 10000 nM T90782 CW7X8B 10866097 EC50 = 2300 nM T90782 C4ND9R 11494976 EC50 = 230 nM T90782 CHB3C7 11510273 Ki > 15000 nM T90782 COI83E 11525909 EC50 > 100000 nM T90782 C9M1FO 11534074 EC50 = 6200 nM T90782 CT74ZJ 11560464 Ki > 15000 nM T90782 CZ8C1X 11606036 EC50 = 2630 nM T90782 CUD1J5 11611428 Ki > 15000 nM T90782 C2XOC1 11993883 EC50 > 1000 nM T90782 COZ6Y2 11993885 EC50 > 100000 nM T90782 CH4XG1 11993887 EC50 > 100000 nM T90782 CZ1J9L 11993889 EC50 > 1000 nM T90782 CQ9ZE4 11993891 EC50 = 120 nM T90782 C3NZ6K 11994005 EC50 > 100000 nM T90782 CNBZ84 11994007 EC50 > 1000 nM T90782 CN0HI1 11994009 EC50 > 1000 nM T90782 CI48FW 11994013 EC50 > 1000 nM T90782 C2MD3V 11995641 EC50 > 100000 nM T90782 CM59TJ 11995643 EC50 > 100000 nM T90782 C4CQ7P 16007361 EC50 = 13 nM T90782 C0R5ZU 16082706 EC50 = 1500 nM T90782 CWK3J0 16082708 EC50 = 3900 nM T90782 C5W8SG 16082709 EC50 = 5500 nM T90782 C7VZA0 16082711 EC50 = 60 nM T90782 CV13PK 16082713 EC50 = 280 nM T90782 C18JCH 16082714 EC50 = 800 nM T90782 C1NV2O 16082716 EC50 = 18000 nM T90782 C6YOF0 16082718 EC50 = 1100 nM T90782 C4FC6S 16082720 EC50 = 4900 nM T90782 C2B6HY 16082731 EC50 = 2500 nM T90782 CG0HJ3 16082734 EC50 = 3500 nM T90782 CD1I6E 16082736 EC50 = 2300 nM T90782 CX5HI6 16082738 EC50 = 560 nM T90782 C31CVA 16082740 EC50 = 1700 nM T90782 CZP86F 16082742 EC50 = 8800 nM T90782 CR6W9O 16216480 EC50 > 20000 nM T90782 CO7FT9 16220889 EC50 > 10000 nM T90782 C3ZEI4 16655024 EC50 > 100000 nM T90782 CIX4T8 22838429 EC50 = 80 nM T90782 C1QCG8 23379800 EC50 = 151 nM T90782 C7GV8K 23662455 IC50 > 10000 nM T90782 CN5OC4 23673110 IC50 = 5300 nM T90782 C20IDU 24857827 EC50 = 1050 nM T90782 C5WP3I 44157464 IC50 = 2550 nM T90782 C6LSQ9 44219765 EC50 = 1900 nM T90782 C3CU9F 44415751 EC50 > 1000 nM T90782 C0SQN9 44415841 EC50 = 230 nM T90782 C9HSG4 44417696 EC50 > 1000 nM T90782 C69SHE 44417704 EC50 > 100000 nM T90782 COZ7M1 44420652 EC50 = 467 nM T90782 CC9VD6 44422901 EC50 > 30000 nM T90782 C2D1MQ 44439743 EC50 > 20000 nM T90782 CW2U7Z 44439757 EC50 > 20000 nM T90782 C42YBU 44439758 EC50 > 20000 nM T90782 C0IBA3 44439765 EC50 > 20000 nM T90782 C1DU4Z 44456078 IC50 > 10000 nM T90782 C1W8IK 44456201 IC50 = 3920 nM T90782 CD50FC 44457390 EC50 = 200 nM T90782 CNW1H5 44457426 EC50 = 18640 nM T90782 C6Z7JE 44457427 EC50 = 20000 nM T90782 CSVR68 44457429 EC50 = 30000 nM T90782 CD5O7G 44583580 IC50 = 10000 nM T90782 C9BM5G 44583581 IC50 > 10000 nM T90782 C84HQM 44585515 EC50 > 10000 nM T90782 C8Q2EX 44585516 EC50 > 10000 nM T90782 C0S8XM 44585517 EC50 > 10000 nM T90782 C1V5YQ 44585518 EC50 = 7830 nM T90782 C9JU8Z 44585519 EC50 = 8190 nM T90782 C09XZT 44585520 EC50 > 10000 nM T90782 CRS2E1 44585521 EC50 > 10000 nM T90782 CTV7A8 44585522 EC50 = 5490 nM T90782 CF3G6K 44585947 EC50 = 610 nM T90782 C7CO0G 44585964 EC50 = 4700 nM T90782 CD9A6E 44585986 EC50 = 5150 nM T90782 CR0W7K 44585987 EC50 = 7700 nM T90782 CUPC35 44585988 EC50 > 10000 nM T90782 CW93JX 44586005 EC50 > 10000 nM T90782 CJHP17 44586025 EC50 = 6830 nM T90782 COB6E3 44586026 EC50 = 6460 nM T90782 CR57TZ 44586027 EC50 = 7330 nM T90782 CV1MB6 44586042 EC50 > 10000 nM T90782 C5JV6T 44586043 EC50 = 8160 nM T90782 C08CEM 44586044 EC50 > 10000 nM T90782 C3R4LJ 44586045 EC50 = 8190 nM T90782 CIA68B 44602426 EC50 >= 100000 nM T90782 CT01NA 44627485 EC50 = 8000 nM T90782 CYP17B 44627487 EC50 = 1990 nM T90782 CL3D1N 44627489 EC50 > 10000 nM T90782 CACW71 44627490 EC50 > 10000 nM T90782 CN9P6R 44627588 EC50 = 10400 nM T90782 CM1R2N 44627590 EC50 > 10000 nM T90782 CN8U1Z 44627592 EC50 = 9100 nM T90782 CGX9A2 44627594 EC50 > 10000 nM T90782 CM3IS5 44627596 EC50 = 1520 nM T90782 CHB4D5 44627598 EC50 > 10000 nM T90782 CD35BV 44627689 EC50 > 10000 nM T90782 CR4CO5 44627691 EC50 > 10000 nM T90782 C7BHI9 44627693 EC50 = 108000 nM T90782 CE6XH9 44627695 EC50 = 2040 nM T90782 CQKW67 44627697 EC50 > 10000 nM T90782 CQ2V9E 44627699 EC50 = 7400 nM T90782 CGT23C 44627801 EC50 = 2760 nM T90782 C5P2FB 44627803 EC50 = 7370 nM T90782 C51QDF 44627805 EC50 > 10000 nM T90782 CCT5S7 45104419 EC50 = 900 nM T90782 CNDO30 45104519 EC50 = 80 nM T90782 CK0L3F 45485232 EC50 = 42 nM T90782 CF6XN5 45485237 EC50 = 127 nM T90782 C12QZE 45485253 EC50 = 3600 nM T90782 C2ZX5J 46232346 EC50 = 47 nM T90782 CNJY69 46232347 EC50 = 140 nM T90782 C18FHS 46232348 EC50 = 230 nM T90782 CJFV20 46830490 EC50 = 1300 nM T90782 CS8I2W 46830491 EC50 = 12 nM T90782 C25PCZ 46830492 EC50 = 63 nM T90782 CK1D4T 46830493 EC50 = 6990 nM T90782 C41UDM 46830782 EC50 > 10000 nM T90782 CT5DY7 46830784 EC50 = 4690 nM T90782 C6BQN5 46830785 EC50 > 10000 nM T90782 C09TMY 46831071 EC50 > 10000 nM T90782 C71DNH 46831072 EC50 = 180 nM T90782 CNR37G 46831073 EC50 = 3490 nM T90782 C2Q0RG 46831384 EC50 = 280 nM T90782 CN26KT 46831386 EC50 = 3510 nM T90782 C0B9RN 46831686 EC50 = 26 nM T90782 CX2Z7P 46831688 EC50 > 10000 nM T90782 CS1D6Q 46831692 EC50 = 80 nM T90782 CJQ84K 46890063 EC50 = 1370 nM T90782 C5S7CK 46890114 EC50 = 2130 nM T90782 CIU19P 46890665 EC50 = 42 nM T90782 CI65GM 46890713 EC50 = 130 nM T90782 C8H5YD 46905555 EC50 = 15 nM T90782 C1WXL6 49861324 EC50 = 70 nM T90782 CPCQ79 51050233 IC50 > 10000 nM T90782 C3XQD5 51050235 IC50 = 4560 nM T90782 CW0N3F 52952183 EC50 = 6100 nM T90782 CK8YW6 52952280 EC50 = 4700 nM T90782 CWR0B6 52952281 EC50 >= 100000 nM T90782 CHC4O2 52952282 EC50 = 6800 nM T90782 CZ86FL 52952283 EC50 = 2500 nM T90782 C2DZ5A 52952391 EC50 = 1370 nM T90782 CA8JY6 52952392 EC50 >= 100000 nM T90782 C2GNH6 52952393 EC50 > 100000 nM T90782 C2IA6G 52952394 EC50 > 100000 nM T90782 C0MWH4 52952395 EC50 > 100000 nM T90782 CZO8K6 52952396 EC50 = 6200 nM T90782 C67NQB 52952397 EC50 > 100000 nM T90782 CBL7S0 52952494 EC50 > 100000 nM T90782 CLGF37 52952495 EC50 = 9800 nM T90782 CA3CS6 52952496 EC50 > 100000 nM T90782 CVO0A1 52952497 EC50 = 142 nM T90782 C15FQS 52952603 EC50 = 8100 nM T90782 CHR9Q8 52952604 EC50 = 1460 nM T90782 C8FUJ5 53262904 EC50 = 950 nM T90782 CA1L7N 53308118 IC50 > 10000 nM T90782 C2JIO7 53308272 EC50 = 230 nM T90782 CDH9J7 53308826 EC50 = 877 nM T90782 CG28DK 53309102 EC50 = 3690 nM T90782 CNLP93 53309244 EC50 = 1170 nM T90782 CYQ90K 53309245 EC50 = 12100 nM T90782 CR3DH9 53309379 EC50 = 4900 nM T90782 C21ZMJ 53309380 EC50 = 5460 nM T90782 CGJ86N 53309381 EC50 = 1650 nM T90782 C4HL7B 53309528 EC50 = 7510 nM T90782 CDN2V9 53309529 EC50 = 1440 nM T90782 CI4G5S 53309530 EC50 = 1640 nM T90782 C4VFI2 68530100 Ki > 15000 nM T90782 CKY3C1 70682678 EC50 = 20110 nM T90782 CUP2I0 70686909 EC50 = 2200 nM T90782 CA0P3V 70688974 EC50 = 8 nM T90782 CQ24UP 70691079 EC50 = 4300 nM T90782 CRF59Q 70691080 EC50 = 60 nM T90782 CNTP42 70691081 EC50 > 10000 nM T90782 CK5QH8 70693210 EC50 = 11230 nM T90782 CMNI96 70695286 EC50 = 200 nM T90782 CTEL13 71459956 EC50 > 100000 nM T90782 CH0O5B 71459957 EC50 > 30000 nM T90782 CF61BN 71459959 EC50 > 30000 nM T90782 CAS84P 76324375 EC50 > 100000 nM T90782 C3P1MQ 90656210 EC50 = 697 nM T90782 C6CEH7 90656211 EC50 = 251 nM T90782 CVOB74 90656212 EC50 = 1780 nM T90782 CL2VA3 90656213 EC50 = 539 nM T90782 C6R2QF 90656214 EC50 = 1210 nM T90782 C6PS8Q 90656215 EC50 = 225 nM T90782 CE32XG 90656216 EC50 = 299 nM T90782 CX53VO 90656217 EC50 = 90 nM T90782 C4W0IB 90656218 EC50 = 9700 nM T90782 C1AD7F 90656219 EC50 = 1330 nM T90782 CL9XR5 90656220 EC50 = 277 nM T90782 C93EMP 90656221 EC50 = 2950 nM T90782 CJ80KG 90656222 EC50 = 4280 nM T90782 CPH41T 90656223 EC50 = 164 nM T90782 CBGQ40 90656224 EC50 = 3000 nM T90782 CA3X6O 90656225 EC50 = 90 nM T90782 C5VWX0 90656226 EC50 = 177 nM T90782 CFCU65 90656227 EC50 = 183 nM T90782 C5FE0D 90656230 EC50 = 23 nM T90782 C4F9RY 90656231 EC50 = 332 nM T90782 C57TEN 90656232 EC50 > 10000 nM T90782 CS7WF2 90666789 EC50 = 39 nM T90782 CE0XU1 90666790 EC50 = 19 nM T90782 C32TOB 90666791 EC50 = 32 nM T90782 CDS2C4 90666792 EC50 = 148 nM T90782 CNV09R 90666793 EC50 = 41 nM T90782 CSE39Z 90666794 EC50 = 100 nM T90782 CG29WU 90666795 EC50 = 9 nM T90782 C40LJI 90666798 EC50 = 126 nM T90782 C58TPX 90666799 EC50 = 731 nM T90782 CGK04R 90666800 EC50 = 1750 nM T90782 CM20EI 90666801 EC50 > 10000 nM T90782 C4HT6U 90666802 EC50 = 879 nM T90782 CM75YG 122185397 EC50 = 203 nM T90782 CVT78Z 122185421 IC50 = 112000 nM T90782 CHIG78 132574706 IC50 = 4360 nM T90782 CA5LF2 135528590 EC50 = 1030 nM T90782 CEA7D5 136169604 IC50 = 69000 nM T90782 C6ZB1D 137632198 IC50 = 4750 nM T90782 C4GA0J 137641946 IC50 > 100000 nM T90782 C7O3US 137643396 IC50 = 12500 nM T90782 CUR8V1 137648798 IC50 = 2670 nM T90782 CR83WH 145978948 EC50 = 12 nM T90782 C3KR0S 145979535 EC50 = 5490 nM T90782 C1VR2K 145981711 EC50 = 493 nM T90782 CJL5U3 145982277 EC50 = 6290 nM T90782 COW27Q 145982347 EC50 = 420 nM T90782 C5EFA6 145984362 EC50 = 705 nM T90782 C2SR0G 145987334 EC50 = 6900 nM T90782 CQA2P7 145988487 EC50 = 4960 nM T90782 C8CHQ3 145989356 EC50 = 2360 nM T90782 C3GDE6 145990456 EC50 = 4120 nM T90782 C68GJS 145990486 EC50 = 49.1 nM T90782 CSV3Q9 145991204 EC50 = 438 nM T90782 C9MLQ6 145991766 EC50 = 47100 nM T90782 CFIO64 145992564 EC50 = 440 nM T90782 CQIS87 145993548 EC50 = 793 nM T90782 C7D9BF 145993852 EC50 = 132 nM T90782 C5LUP8 155516521 EC50 > 3000 nM T90782 CT83QU 155540535 EC50 = 1390 nM T90782 C6MG8A 90656228 EC50 = 334 nM T90782 D01ZZJ 49867142 EC50 > 100000 nM T90782 D02HAL 6031 EC50 = 13 nM T90782 D03WBX 44585949 EC50 = 339 nM T90782 D03YRN 16078986 IC50 = 37 nM T90782 D04IWB 10174453 EC50 > 1000 nM T90782 D05MXI 42611190 IC50 > 10000 nM T90782 D05NWF 6022 EC50 = 65000 nM T90782 D06PIW 53262902 EC50 = 740 nM T90782 D07LYU 53262890 EC50 = 1210 nM T90782 D07MIE 8629 EC50 = 1600 nM T90782 D07MTB 11510579 Ki > 15000 nM T90782 D07TSE 16082712 EC50 = 447 nM T90782 D07XZT 6132 EC50 = 88000 nM T90782 D08DXA 23675622 IC50 = 2790 nM T90782 D08VPN 22960366 EC50 = 28 nM T90782 D0B0ZQ 9875920 IC50 = 4340 nM T90782 D0C7LS 135398619 EC50 = 45000 nM T90782 D0P0EP 161647 EC50 > 100000 nM T90782 D0P4GP 52952605 EC50 = 7000 nM T90782 D0P6KN 44457307 EC50 = 154 nM T90782 D0P7RI 9872620 EC50 = 291 nM T90782 D0Q1HE 16116566 EC50 > 10000 nM T90782 D0RV7M 145729 EC50 = 1720 nM T90782 D0T4WF 11994011 EC50 = 70 nM T90782 D0U1OJ 5310983 EC50 = 100000 nM T02546 D03FLC 3878 Ki = 17000 nM T02546 D04MSM 2554 Ki = 52000 nM T02546 D0C7ET 11174599 IC50 = 7.6 nM T02546 D0E4DW 1775 Ki = 24000 nM T02546 D0UM7O 3821 IC50 = 2300000 nM T02546 D0X4RN 3676 IC50 = 2000 nM T02546 D00BUR 216327 IC50 > 1000 nM T02546 D0K9IF 71666749 IC50 > 30000 nM T02546 D0O7QA 46840946 IC50 = 10000 nM T02546 D0OX9F 16046068 IC50 = 10000 nM T02546 D07EQF 9816959 Ki = 180 nM T02546 C0DSE7 17155 Ki = 61000 nM T02546 C7D8TC 185376 EC50 = 26915.35 nM T02546 CXL10N 599984 Ki = 81000 nM T02546 CR4G2M 643321 EC50 = 208929.61 nM T02546 CPN25U 998021 IC50 = 10000 nM T02546 CG70HP 3080825 EC50 = 275422.87 nM T02546 C7M3QH 3080827 EC50 = 223872.11 nM T02546 CFN3Z8 6603917 EC50 = 5754.4 nM T02546 C61YOH 6950526 EC50 = 234422.88 nM T02546 CP9I0X 9818665 Ki = 31 nM T02546 CZ3OX8 9861009 Ki = 31 nM T02546 CX38SK 9948785 Ki = 25 nM T02546 C01LUV 10353340 EC50 = 12022.64 nM T02546 C3XN2T 10377047 EC50 = 3019.95 nM T02546 CU5O3A 10442602 EC50 = 23442.29 nM T02546 CR49JY 10537392 EC50 = 17378.01 nM T02546 C70QGH 10609631 EC50 = 67608.3 nM T02546 C3PJQ6 10634184 EC50 = 501187.23 nM T02546 CH8EN7 10637348 EC50 = 2398.83 nM T02546 C36QIC 10681102 EC50 = 67608.3 nM T02546 CMDO50 10752970 EC50 = 199526.23 nM T02546 C0GDA1 10823492 EC50 = 28183.83 nM T02546 C16FKH 10846493 EC50 = 40738.03 nM T02546 CGE4I0 10847196 EC50 = 218776.16 nM T02546 C5Y2GT 11150055 EC50 = 7943.28 nM T02546 CX8A9W 11184951 EC50 = 19498.45 nM T02546 CH3X2Z 11198140 Ki = 340 nM T02546 C2GDL6 11242617 Ki = 690 nM T02546 CI7NC8 11253662 EC50 = 10000 nM T02546 C7TR2B 11300443 Ki = 35 nM T02546 CE4D6X 11391352 EC50 = 15135.61 nM T02546 CY2HZ1 11459294 EC50 = 3019.95 nM T02546 C16LPK 11738446 Ki = 150 nM T02546 CS0M5W 14796880 EC50 = 3019.95 nM T02546 CUZ0K4 17757962 EC50 = 1698.24 nM T02546 CF3E9I 17758080 EC50 = 2290.87 nM T02546 CL73HJ 21589240 IC50 = 0.062 nM T02546 C8X9SG 25058834 EC50 = 1000 nM T02546 CPRA85 25793315 EC50 = 3981.07 nM T02546 CDG3Z4 25793317 EC50 = 15848.93 nM T02546 CU12YJ 44593012 EC50 = 31622.78 nM T02546 C4C8PF 44593013 EC50 = 10000 nM T02546 CV5F2S 44593027 EC50 = 501187.23 nM T02546 C6QF4X 44593029 EC50 = 5754.4 nM T02546 C9V6FI 44593042 EC50 = 3715.35 nM T02546 CQ37SU 44593043 EC50 = 2884.03 nM T02546 CAHE37 44593075 EC50 = 7079.46 nM T02546 C98NKD 44593076 EC50 = 4677.35 nM T02546 CK5QG1 44593077 EC50 = 2691.53 nM T02546 CU9BT2 44593078 EC50 = 1905.46 nM T02546 CSD09H 44593334 EC50 = 11220.18 nM T02546 C8YXN7 44593335 EC50 = 9120.11 nM T02546 CS5EJ1 46841648 IC50 > 10000 nM T02546 CRE97F 46841787 IC50 > 30000 nM T02546 C06OXV 52920492 IC50 = 24000 nM T02546 CMS2F7 53239561 IC50 = 4580 nM T02546 C23WVS 53361524 IC50 = 400 nM T02546 CYF3R7 60167367 IC50 = 14000 nM T02546 C2MC6B 71522734 IC50 > 10000 nM T02546 C7OE1X 76309796 IC50 = 16000 nM T02546 CBH4N7 76309797 IC50 > 30000 nM T02546 C10UTF 76310404 IC50 > 30000 nM T02546 C6T1NV 76310406 IC50 > 30000 nM T02546 CC4BK5 76310408 IC50 > 30000 nM T02546 C8M7RN 76310409 IC50 > 30000 nM T02546 CHFC49 76313502 IC50 > 30000 nM T02546 C1PM7H 76314065 IC50 > 30000 nM T02546 CBK0T8 76314067 IC50 > 30000 nM T02546 C20ILA 76314069 IC50 = 28000 nM T02546 C8OQT1 76314070 IC50 > 30000 nM T02546 CNM4K0 76317019 IC50 = 16000 nM T02546 C32OSF 76317020 IC50 > 30000 nM T02546 CKG5A9 76317629 IC50 > 30000 nM T02546 CQ7JK4 76317631 IC50 > 30000 nM T02546 CT2R5J 76320732 IC50 = 8000 nM T02546 CVP8U9 76320733 IC50 = 30000 nM T02546 C2RJW0 76320734 IC50 = 15000 nM T02546 CY8NT4 76321352 IC50 > 30000 nM T02546 CRU30A 76321353 IC50 > 30000 nM T02546 C46MFT 76324385 IC50 = 21000 nM T02546 C4W1NV 76324386 IC50 > 30000 nM T02546 CJF20G 76324950 IC50 = 26000 nM T02546 CP3UI7 76327945 IC50 > 30000 nM T02546 CNY5X1 76328517 IC50 > 30000 nM T02546 CX54MA 76328518 IC50 = 25000 nM T02546 CINA95 76331591 IC50 > 30000 nM T02546 CCXK29 76332197 IC50 > 30000 nM T02546 CH4K7Q 76332198 IC50 = 15000 nM T02546 C4WO6Y 76332199 IC50 > 30000 nM T02546 CK47NO 76332200 IC50 > 30000 nM T02546 CANB89 76332201 IC50 > 30000 nM T02546 CO2N7R 76335221 IC50 = 25000 nM T02546 C05RSQ 76335223 IC50 > 30000 nM T02546 C8ND6L 76335224 IC50 > 30000 nM T02546 CUO84S 76335833 IC50 > 30000 nM T02546 CTG76E 86687532 IC50 = 17000 nM T02546 CC5N9I 117737142 IC50 > 14000 nM T02546 C10BKY 117749324 IC50 > 42500 nM T02546 C9KV7L 117993993 IC50 = 1100 nM T02546 C7AYV5 118540795 IC50 = 1451 nM T02546 CR8TX9 118708662 IC50 = 30 nM T02546 C69PLO 118734433 IC50 > 4800 nM T02546 C2NAE8 118734434 IC50 = 1800 nM T02546 CD4B5E 118734435 IC50 > 3000 nM T02546 C91PCO 118734436 IC50 = 3200 nM T02546 CM2Y6W 118734437 IC50 = 8500 nM T02546 CFL60J 118734438 IC50 = 3800 nM T02546 CQ0R3E 118734439 IC50 > 4600 nM T02546 CY8A1T 118734440 IC50 > 3900 nM T02546 CFRZ45 118734441 IC50 = 3000 nM T02546 C3ZJ0K 118734442 IC50 = 3000 nM T02546 CI30YK 118734443 IC50 = 900 nM T02546 CUAQ60 118734444 IC50 = 2700 nM T02546 CFNR84 118734445 IC50 = 4700 nM T02546 CK12TX 118734446 IC50 = 3000 nM T02546 C09BDT 118734447 IC50 = 1500 nM T02546 C6F9BI 118734448 IC50 > 5000 nM T02546 C8ZLX9 118734449 IC50 = 3000 nM T02546 C01BNE 118734450 IC50 = 3700 nM T02546 CI0FE2 118734451 IC50 = 1900 nM T02546 C1CED0 118734452 IC50 > 5000 nM T02546 C8NBL5 118734453 IC50 = 3200 nM T02546 C0CY2K 118734454 IC50 = 4100 nM T02546 CTR7O8 118734455 IC50 > 4900 nM T02546 CZQD84 118734456 IC50 > 4500 nM T02546 CGBF25 118734457 IC50 > 5000 nM T02546 C6I8HF 118734458 IC50 > 5000 nM T02546 C5G7DQ 118734459 IC50 = 4500 nM T02546 CVW15D 118734460 IC50 > 5000 nM T02546 CSE60C 118734461 IC50 > 5000 nM T02546 CO4U1R 118734462 IC50 = 11000 nM T02546 CA95IF 118734463 IC50 > 10000 nM T02546 C14ILF 118734464 IC50 = 4600 nM T02546 C3TOV9 118734465 IC50 = 4100 nM T02546 C2RO8T 118734466 IC50 = 900 nM T02546 CSP25D 118734467 IC50 = 2000 nM T02546 CJD80C 118734468 IC50 = 900 nM T02546 C06TAI 118734469 IC50 = 7700 nM T02546 CBY5M0 118734470 IC50 = 4700 nM T02546 CHO8I3 118734471 IC50 = 100 nM T02546 C38BCH 118734472 IC50 = 1700 nM T02546 CV7UH5 118734473 IC50 = 1500 nM T02546 C6SEA7 118734474 IC50 = 1100 nM T02546 CO7DP2 118734475 IC50 = 100 nM T02546 CX2R0E 118734476 IC50 = 70 nM T02546 C16AEK 118734477 IC50 = 410 nM T02546 CO1UF9 118734478 IC50 = 90 nM T02546 C16AUM 118734479 IC50 = 140 nM T02546 CI2P1V 118734480 IC50 = 3400 nM T02546 C1Z8AN 118734481 IC50 = 240 nM T02546 CYD8N6 118734482 IC50 = 110 nM T02546 CW05LY 118734483 IC50 = 2600 nM T02546 CN01US 118734484 IC50 = 9900 nM T02546 C3E7GP 118734485 IC50 = 740 nM T02546 CCA41Z 118734486 IC50 = 6100 nM T02546 CM2QS5 118734487 IC50 = 500 nM T02546 C3T1QC 118734488 IC50 = 530 nM T02546 CM6Y8X 118734489 IC50 = 110 nM T02546 C93LMC 118734490 IC50 = 4900 nM T02546 C8LHA3 118734491 IC50 = 240 nM T02546 C26ADB 118734547 IC50 = 2800 nM T02546 C82UBF 118734548 IC50 > 5000 nM T02546 CO4KD2 118734549 IC50 > 10000 nM T02546 CX6L4C 118734550 IC50 = 1200 nM T02546 C5JNX2 118734551 IC50 = 3300 nM T02546 C0UJ8Q 118734552 IC50 = 6600 nM T02546 CJDP52 118734553 IC50 = 1900 nM T02546 C9Q2ND 121333973 IC50 = 12000 nM T02546 C7JT8V 127045799 IC50 = 210 nM T02546 CH2Z3S 127045806 IC50 = 2400 nM T02546 CSJD60 127045808 IC50 = 4000 nM T02546 COWD91 127045811 IC50 > 5000 nM T02546 C90JPN 127045813 IC50 > 5000 nM T02546 C21JCE 127045825 IC50 > 5000 nM T02546 CNF0G1 127045829 IC50 > 5000 nM T02546 CC9TY3 127045830 IC50 = 1500 nM T02546 CDC0M9 127046018 IC50 = 1200 nM T02546 C74SHI 127046022 IC50 = 3900 nM T02546 CH0CD1 127046023 IC50 > 4900 nM T02546 CPX1F0 127046025 IC50 > 5000 nM T02546 CAVD37 127046026 IC50 > 4000 nM T02546 C8UW6X 127046032 IC50 = 600 nM T02546 CMPZ51 127046033 IC50 = 600 nM T02546 CY5J0R 127046039 IC50 = 2600 nM T02546 CBQ47D 127046045 IC50 = 3700 nM T02546 C6NVQ1 127046047 IC50 > 4600 nM T02546 C4MU2J 127046230 IC50 = 2600 nM T02546 CGYE23 127046231 IC50 > 5000 nM T02546 C69GBJ 127046239 IC50 = 2000 nM T02546 CM1IH3 127046241 IC50 = 1800 nM T02546 C4L1VA 127046242 IC50 = 2600 nM T02546 CWN2J7 127046243 IC50 = 550 nM T02546 CI1VA2 127046252 IC50 = 3800 nM T02546 CE67AD 127046253 IC50 = 70 nM T02546 C53RIX 127046257 IC50 = 4100 nM T02546 COK9Z3 127046259 IC50 = 1400 nM T02546 CL5VY9 127046359 IC50 = 170 nM T02546 C3M6YT 127046415 IC50 = 2900 nM T02546 C90HYR 127046420 IC50 = 2000 nM T02546 C8BES0 127046422 IC50 = 720 nM T02546 C2EI4Q 127046423 IC50 = 13000 nM T02546 CM2HB0 127046424 IC50 = 900 nM T02546 CM5D6J 127046425 IC50 = 500 nM T02546 C9LH4U 127046428 IC50 > 5000 nM T02546 C20KGH 127046429 IC50 = 2000 nM T02546 CH27MP 127046433 IC50 > 5000 nM T02546 CWH7Y0 127046434 IC50 > 5000 nM T02546 C1CV8E 127046436 IC50 = 2500 nM T02546 C87YLU 127046583 IC50 > 5000 nM T02546 C74ELB 127046587 IC50 = 400 nM T02546 CI9XY7 127046589 IC50 = 2300 nM T02546 CQ3EV4 127046592 IC50 = 1700 nM T02546 C8PO4C 127046597 IC50 = 4400 nM T02546 C31XHN 127046598 IC50 = 700 nM T02546 CFSH84 127046606 IC50 = 1900 nM T02546 CP8T2D 127046764 IC50 = 700 nM T02546 C0A7SK 127046767 IC50 > 5000 nM T02546 CC2Y1J 127046770 IC50 > 5000 nM T02546 C1XON9 127046774 IC50 > 5000 nM T02546 C80RLU 127046781 IC50 > 5000 nM T02546 CSKX63 127046908 IC50 = 1300 nM T02546 CVUW94 127046909 IC50 = 3400 nM T02546 C02HPV 127046912 IC50 = 2000 nM T02546 C8CK6P 127046914 IC50 > 5000 nM T02546 C3CSI0 127046916 IC50 = 160 nM T02546 C4X2OU 127046919 IC50 = 3200 nM T02546 CL9W8T 127046920 IC50 = 400 nM T02546 CLH51Y 127046923 IC50 > 5000 nM T02546 CXMC23 127046930 IC50 > 5000 nM T02546 CB9EF5 127046932 IC50 = 600 nM T02546 CZ7G6T 127047057 IC50 = 2300 nM T02546 CND20E 127047062 IC50 = 1500 nM T02546 CNSZ83 127047063 IC50 > 2200 nM T02546 C1R4VN 127047068 IC50 > 5000 nM T02546 C5VU7H 127047069 IC50 = 2200 nM T02546 CFG94A 127047073 IC50 > 5000 nM T02546 CF5D0S 127047074 IC50 > 5000 nM T02546 C0XS7B 127047075 IC50 > 5000 nM T02546 CI60KD 127047206 IC50 = 2100 nM T02546 CA7YG4 127047208 IC50 > 5000 nM T02546 CXT5Y0 127047216 IC50 = 1100 nM T02546 CY8RH9 127047220 IC50 > 5000 nM T02546 CV4OB1 127047223 IC50 = 3900 nM T02546 CFPJ73 127047320 IC50 > 5000 nM T02546 C3JK6P 127047322 IC50 = 2600 nM T02546 C1T5PC 127047323 IC50 = 1300 nM T02546 C28REX 127047327 IC50 = 1100 nM T02546 CVSF19 127047330 IC50 > 5000 nM T02546 C0IO2K 127047331 IC50 = 2300 nM T02546 C9SIK3 127047333 IC50 = 1400 nM T02546 CKD78E 127047346 IC50 = 700 nM T02546 C5DO7I 127047347 IC50 = 1500 nM T02546 CM5TX2 127047468 IC50 > 5000 nM T02546 C54TRJ 127047469 IC50 = 1400 nM T02546 C3K5YI 127047471 IC50 = 3500 nM T02546 C2M5JH 127047472 IC50 = 900 nM T02546 C3SLJ4 127047473 IC50 = 500 nM T02546 CCA51M 127047474 IC50 = 2300 nM T02546 C6EM0G 127047476 IC50 > 5000 nM T02546 C5RKB7 127047479 IC50 = 700 nM T02546 C96VDX 127047480 IC50 = 2400 nM T02546 CJ7IQ4 127047485 IC50 = 500 nM T02546 CZKB91 127047487 IC50 = 4400 nM T02546 C7OTX3 127047488 IC50 = 1500 nM T02546 CVR95B 127047489 IC50 = 1000 nM T02546 CW8P5Y 127047613 IC50 = 2400 nM T02546 C0WXP3 127047615 IC50 = 1770 nM T02546 C1RK5C 127047619 IC50 > 5000 nM T02546 C9QZH7 127047622 IC50 = 290 nM T02546 CJ31BC 127047628 IC50 > 5000 nM T02546 C9MXK5 127047633 IC50 = 600 nM T02546 C1ULZ3 127047735 IC50 > 3800 nM T02546 C4T5WS 127047736 IC50 > 5000 nM T02546 CQ45AO 127047757 IC50 > 4100 nM T02546 CG5X0Y 127047758 IC50 = 1400 nM T02546 CTRE63 127047854 IC50 > 5000 nM T02546 CDGS14 127047866 IC50 > 5000 nM T02546 C16NUB 127047867 IC50 = 2300 nM T02546 CG52RP 127047873 IC50 = 4400 nM T02546 C8PWL6 127047983 IC50 > 5000 nM T02546 CGW63M 127047988 IC50 = 700 nM T02546 CR6AB0 127047989 IC50 > 5000 nM T02546 CK9ZO8 127047990 IC50 = 2500 nM T02546 CQ2SO8 127047999 IC50 = 730 nM T02546 C2D9LN 127048108 IC50 = 1400 nM T02546 C25GJD 127048113 IC50 = 200 nM T02546 C4VID9 127048115 IC50 > 4900 nM T02546 CCI81A 127048120 IC50 > 5000 nM T02546 CE1Z4W 127048121 IC50 = 3100 nM T02546 CI0P1M 127048127 IC50 = 1500 nM T02546 C4CUP9 127048128 IC50 = 700 nM T02546 C7HGD0 127048130 IC50 = 420 nM T02546 C4LK6A 127048137 IC50 > 5000 nM T02546 CNA30T 127048138 IC50 = 750 nM T02546 CZ5H2B 132020452 IC50 = 4800 nM T02546 C04JSE 137649716 IC50 = 4000 nM T02546 CR23HX 145948497 IC50 = 3900 nM T02546 CNSU46 145948687 IC50 > 4800 nM T02546 CRH94T 145948711 IC50 > 3000 nM T02546 CDZK19 145948712 IC50 = 2600 nM T02546 C8KW9F 145948730 IC50 = 650 nM T02546 CQPL31 145948977 IC50 > 5000 nM T02546 C5K7VF 145950190 IC50 = 72 nM T02546 C3IPL7 145951679 IC50 = 117 nM T02546 C23NCA 145951748 IC50 = 23 nM T02546 CCR2Y5 145952753 IC50 = 102 nM T02546 CHV56N 145953458 IC50 = 258 nM T02546 CRT63U 145953831 IC50 = 182 nM T02546 CF6L8Q 145955101 IC50 = 53 nM T02546 CSX5K2 145955231 IC50 = 37 nM T02546 CTW9Q4 145956356 IC50 = 23 nM T02546 C8NH1M 145957393 IC50 = 39 nM T02546 CL59SC 145958162 IC50 = 52 nM T02546 CVX4N1 145958248 IC50 = 92 nM T02546 CCTB54 145958837 IC50 = 104 nM T02546 C38DYW 145959291 IC50 = 145 nM T02546 CDW83O 145959527 IC50 = 89 nM T02546 CHX92D 145960265 IC50 = 162 nM T02546 CSK8Y1 145965486 IC50 = 2900 nM T02546 COS4B9 145972887 IC50 = 193 nM T02546 C5UE1S 145973817 IC50 = 177 nM T02546 CUV49K 145977796 IC50 = 25200 nM T02546 COZ54G 155523716 IC50 = 5300 nM T02546 C5F9BQ 155526497 IC50 = 75000 nM T02546 CEL05R 155543885 IC50 = 20 nM T02546 CE3H4Z 155567528 IC50 = 140 nM T02546 CH8Z4R 44593058 EC50 = 22908.68 nM T02546 C2E5CL 44593059 EC50 = 3019.95 nM T02546 D03NLL 180621 EC50 = 22908.68 nM T02546 D0KH1D 9816478 Ki = 200 nM T02546 D0M5VF 2806138 Ki = 240 nM T02546 D0P8TL 56947150 IC50 = 19 nM T91113 D0R1RS 3715 IC50 > 100000 nM T91113 C7WBY9 10079225 IC50 = 4.2 nM T91113 CL0M1W 10652466 IC50 = 165 nM T91113 D0HD9P 444899 IC50 > 100000 nM T91113 D0J8TY 5280436 IC50 = 420 nM T36729 C0HT3G 1014304 IC50 = 25000 nM T36729 C4SED3 1226613 IC50 = 40000 nM T36729 CQ21NS 4112136 Ki = 4720 nM T36729 C7AZ5R 7233583 IC50 > 100000 nM T36729 CH28EJ 51035513 Ki = 645 nM T36729 C7OB2X 51035721 Ki = 1340 nM T36729 C3AH5R 51035722 Ki = 1160 nM T36729 CL96PR 51035723 Ki = 1195 nM T36729 C56YLK 51035724 Ki = 1150 nM T36729 CL2CN8 51035725 Ki = 365 nM T36729 C4LK5D 51035726 Ki = 1280 nM T36729 C3H1VJ 51035928 Ki = 1260 nM T36729 C91XOM 51035929 Ki = 1760 nM T36729 C6U2YK 51035930 Ki = 780 nM T36729 C26PCE 51035931 Ki = 1020 nM T36729 C42XGB 51035932 Ki = 2015 nM T36729 CF8C6B 51036143 Ki = 510 nM T36729 C9B2SY 51036144 Ki = 820 nM T36729 CU04RE 51036146 Ki = 1370 nM T36729 C1YQ7L 57395836 Ki = 1140 nM T36729 C25RKI 57395837 Ki = 433 nM T36729 C8LUQ1 86301661 IC50 = 9000 nM T36729 CD0E3K 118718001 IC50 = 31000 nM T36729 C93NJU 118718002 IC50 = 30000 nM T36729 C1EYV6 118718011 IC50 > 100000 nM T36729 CNSL51 118718012 IC50 > 100000 nM T36729 C8C5BD 118718020 IC50 = 40000 nM T36729 CT6K9C 118718021 IC50 = 12000 nM T36729 CJF9B1 118718025 IC50 = 51000 nM T36729 C49APK 118718026 IC50 = 20000 nM T36729 C2UTX3 118718027 IC50 = 30 nM T36729 CS56VP 118718039 IC50 > 100000 nM T36729 C8OJX0 118718040 IC50 = 79000 nM T36729 CST27I 118718052 IC50 = 27000 nM T36729 CYU08F 118718053 IC50 > 100000 nM T36729 D06UEP 17027464 Ki = 1530 nM T30219 CAH5N0 5490359 EC50 = 3800 nM T30219 C05BAM 9961381 IC50 = 27000 nM T30219 CRK13Y 10486513 EC50 = 199.53 nM T30219 CFY65T 10725013 EC50 = 5700 nM T30219 CWL03J 17753143 IC50 = 50.12 nM T30219 C7LR8V 17753265 IC50 = 79.43 nM T30219 C9ATW3 24829327 IC50 = 50 nM T30219 CK45HA 25156014 IC50 = 3.981 nM T30219 C5MP6R 44426457 IC50 = 316.23 nM T30219 C5AQE0 44426458 IC50 = 125.89 nM T30219 CZN62U 44426459 IC50 = 316.23 nM T30219 CFM04J 44426460 IC50 = 199.53 nM T30219 C2M6OU 44426461 IC50 = 794.33 nM T30219 CVZU84 44426462 IC50 = 199.53 nM T30219 C9Z0DU 44426463 EC50 = 501.19 nM T30219 C9J5TU 44426464 IC50 = 199.53 nM T30219 C5ON4Y 44426465 IC50 = 794.33 nM T30219 C1ABZ5 44426466 IC50 = 1584.89 nM T30219 C95MVL 44426469 IC50 = 316.23 nM T30219 C29ACK 44426470 IC50 = 3981.07 nM T30219 CRMQ72 44426471 IC50 = 100000 nM T30219 CTG6X3 44426472 IC50 = 794.33 nM T30219 C0D4FE 44426475 IC50 = 6309.57 nM T30219 C8Y4BS 44426478 IC50 = 50118.72 nM T30219 CUG1H3 44426481 IC50 = 794.33 nM T30219 CB12JM 44426495 IC50 = 31.62 nM T30219 CI4PX8 44426496 IC50 = 15.85 nM T30219 CZJ87Q 44426497 EC50 = 125.89 nM T30219 CHJ20D 44430510 IC50 = 630.96 nM T30219 CJ69LC 44430513 IC50 = 79432.82 nM T30219 CW7XF5 44430514 IC50 = 3162.28 nM T30219 CJ9T2Y 44430516 IC50 = 19952.62 nM T30219 CYE82D 44430519 IC50 = 316.23 nM T30219 C9IH2L 44430526 IC50 = 1000 nM T30219 CLOP76 44430527 IC50 = 630.96 nM T30219 C93BJH 44430528 IC50 = 63095.73 nM T30219 C7PWR2 44430529 IC50 = 25118.86 nM T30219 CM92EX 44430530 IC50 = 794.33 nM T30219 CX3OZ2 44430531 IC50 = 794.33 nM T30219 CK35BF 44430532 IC50 = 3162.28 nM T30219 CY6AX7 44430533 IC50 = 794.33 nM T30219 C5ZKM0 44430536 IC50 = 2511.89 nM T30219 CJ34QT 44430538 IC50 = 125.89 nM T30219 CJ5C3Q 44430539 IC50 = 630.96 nM T30219 C3D2WP 44430541 IC50 = 199.53 nM T30219 C3UOE2 44430546 IC50 = 1995.26 nM T30219 CA5SG0 44430547 EC50 = 199.53 nM T30219 CJL87C 44430548 IC50 = 158.49 nM T30219 C7BF5P 44430549 IC50 = 100 nM T30219 CMH04P 44430550 IC50 = 316.23 nM T30219 CLU0A4 44430551 EC50 = 1584.89 nM T30219 CLS05Y 44430552 IC50 = 1000 nM T30219 C7N0GA 44430553 IC50 = 15848.93 nM T30219 C50GXV 44430554 EC50 = 199.53 nM T30219 C1M6BT 44430555 IC50 = 1258.93 nM T30219 C2FTZ9 44430556 IC50 = 1000 nM T30219 CE1N0R 44430557 IC50 = 50118.72 nM T30219 C2Q4ZH 44430558 IC50 = 1995.26 nM T30219 CQA74Z 44430559 IC50 = 10000 nM T30219 CZ14RV 44430560 IC50 = 12589.25 nM T30219 C8AB0N 44431783 IC50 = 199.53 nM T30219 CV6Y2P 45263542 IC50 = 5011.87 nM T30219 CRGO95 46855352 EC50 = 1995.26 nM T30219 C5AN9E 46855353 EC50 = 1800 nM T30219 C09CKZ 46855354 EC50 = 780 nM T30219 C4Z1FN 46855499 EC50 = 38000 nM T30219 CCV7R8 46855634 EC50 = 309.03 nM T30219 C5NE7X 46855776 EC50 = 2630.27 nM T30219 CK1P9F 46855777 IC50 = 240 nM T30219 C40YFU 46911378 IC50 = 82 nM T30219 CN5R3O 46911429 IC50 = 41.69 nM T30219 CW78DI 49799080 IC50 = 251.19 nM T30219 C8PH3O 49799081 IC50 = 12.59 nM T30219 CO48HR 49799082 IC50 = 740 nM T30219 C1QE2Y 49799083 IC50 = 6300 nM T30219 CH74LZ 49799085 EC50 = 31622.78 nM T30219 C4VY3M 49799092 EC50 = 950 nM T30219 C8Z3UG 49799093 EC50 = 398.11 nM T30219 CCNM89 49799094 EC50 = 5011.87 nM T30219 CHZ91Y 49799095 EC50 = 5011.87 nM T30219 CFHK40 49799096 EC50 = 1000 nM T30219 CS5BD9 49799097 IC50 = 275.42 nM T30219 CH1CS0 49799098 EC50 = 720 nM T30219 CZ8P3Q 49799099 EC50 = 3800 nM T30219 C8T3OZ 49799104 EC50 = 25000 nM T30219 CFSY26 49799105 IC50 = 244 nM T30219 CT69GA 49799106 EC50 = 10964.78 nM T30219 CC6FG0 49799107 EC50 = 520 nM T30219 CY76HG 49799139 EC50 = 2454.71 nM T30219 CHB6T4 49799142 EC50 = 6760.83 nM T30219 CLNQ20 49799143 IC50 = 166 nM T30219 C3J2FE 49799144 EC50 = 467.74 nM T30219 CPD82O 49799145 EC50 = 1174.9 nM T30219 CHT25O 49799146 EC50 = 489.78 nM T30219 CRJD42 49799147 EC50 = 512.86 nM T30219 C1OC4V 49799148 EC50 = 1096.48 nM T30219 COR0Z4 49799149 EC50 = 354.81 nM T30219 C0DHW9 49799151 IC50 = 8200 nM T30219 C4NT3M 49799153 EC50 = 28840.32 nM T30219 CKV60X 49799155 EC50 = 36307.81 nM T30219 C52YFU 70687669 EC50 = 57000 nM T30219 CU2N9Y 71525749 IC50 = 5 nM T30219 CX03AW 71565506 EC50 = 72.44 nM T30219 CCXZ27 71565508 IC50 = 794.33 nM T30219 C81WQO 71565509 IC50 = 157 nM T30219 CKJ12C 71565510 IC50 = 54.95 nM T30219 C3ZLX6 71565580 EC50 = 7.586 nM T30219 CQ8XU0 71565581 IC50 = 141.25 nM T30219 C58ZDQ 71565582 EC50 = 54 nM T30219 CU31AW 71566580 IC50 = 19 nM T30219 CHEN47 71566581 EC50 = 26.92 nM T30219 C8YN4U 71566652 IC50 = 27 nM T30219 C06ZFN 71566653 IC50 = 137 nM T30219 C71NEF 71566654 EC50 = 7 nM T30219 CUY9D2 71768012 EC50 = 19 nM T30219 CWA98J 89570147 IC50 = 1144 nM T30219 C30ANF 89570392 IC50 = 104 nM T30219 CLS1X2 89570442 IC50 = 10 nM T30219 CLA4M3 89570463 IC50 = 87 nM T30219 C7PA4X 89570464 IC50 = 600 nM T30219 C3W8NR 101886248 IC50 = 6.31 nM T30219 CS5BG0 101886249 IC50 = 50.12 nM T30219 CZHX76 101886250 IC50 = 31 nM T30219 C3J9AN 101886251 IC50 = 2900 nM T30219 CWI1D6 101886252 IC50 = 100 nM T30219 C5DV8G 101886253 IC50 = 4 nM T30219 C9GFU6 101886254 IC50 = 12 nM T30219 CB9TS3 117634949 IC50 = 707.95 nM T30219 CCK4P7 117634952 IC50 = 102 nM T30219 CB7D1N 117634979 EC50 = 740 nM T30219 CK2DA8 117634981 IC50 = 967 nM T30219 C7PMW6 117637102 EC50 = 850 nM T30219 C1GZ4S 118716617 IC50 = 100 nM T30219 CMA04D 122392665 EC50 = 15 nM T30219 CFL40V 122392666 IC50 = 320 nM T30219 C56MWH 127034742 IC50 = 446.68 nM T30219 CS7UA2 127034743 IC50 = 1023.29 nM T30219 CQ3NB4 127034744 EC50 = 45 nM T30219 C8VT3Z 127035774 IC50 = 1300 nM T30219 CIU3C5 127036518 EC50 = 40.74 nM T30219 CN5TX7 135418443 IC50 = 1700 nM T30219 C4ECV2 136110886 IC50 = 11410 nM T30219 C7JR9W 136110887 IC50 = 5970 nM T30219 CF4DT8 136110888 IC50 = 8450 nM T30219 CPO60R 136110889 IC50 = 7160 nM T30219 CSM8X6 136110890 IC50 = 12550 nM T30219 CFMN09 136110891 IC50 = 6140 nM T30219 CV84AG 136110892 IC50 = 5900 nM T30219 C5Y4VR 136110893 IC50 = 5360 nM T30219 C3APK0 136110894 IC50 = 48000 nM T30219 COE2I9 136110895 IC50 = 32000 nM T30219 CPM36X 136110896 IC50 = 13400 nM T30219 C4F3EP 136110897 IC50 = 7480 nM T30219 CASR54 145996525 IC50 = 10 nM T30219 C8ZGW5 155510486 IC50 = 3.981 nM T30219 C9KEZ6 155513738 IC50 > 10000 nM T30219 C96JTL 155516924 IC50 = 1995.26 nM T30219 C10PAL 155518058 IC50 = 3 nM T30219 C8LKQ2 155525092 IC50 = 100 nM T30219 C6Q9ZD 155526496 IC50 = 200 nM T30219 CQ8WY7 155527368 EC50 = 50 nM T30219 CZF9G2 155534229 IC50 = 790 nM T30219 CJN86Y 155534696 IC50 = 1.995 nM T30219 C6EQ5J 155535658 IC50 = 6100 nM T30219 COJE04 155535683 IC50 = 140 nM T30219 C5M6JX 155535693 IC50 = 100 nM T30219 CM8PE3 155536326 IC50 = 31.62 nM T30219 C3ZV4U 155541887 EC50 > 100000 nM T30219 C76YCF 155542585 IC50 > 10000 nM T30219 CHLK68 155546129 IC50 = 2300 nM T30219 CN4IS7 155554899 IC50 = 125.89 nM T30219 C9RI1A 155555271 IC50 = 2400 nM T30219 CVP5N7 155557086 EC50 > 100000 nM T30219 C07QEB 155557328 IC50 = 31.62 nM T30219 C78NEJ 155557799 IC50 = 39.81 nM T30219 CHXF78 155558856 IC50 = 100 nM T30219 CJ6KF1 155563876 IC50 = 3981.07 nM T30219 CU0KN2 155569071 EC50 = 100000 nM T30219 D01OIJ 91827354 IC50 = 10 nM T30219 D01QQD 91827355 IC50 = 794.33 nM T30219 D0S8NM 5311120 IC50 = 1.3 nM T12091 D07HPJ 11476171 IC50 = 2900 nM T12091 D0E3TC 44259 IC50 = 10005 nM T12091 D0MR0B 54766013 IC50 > 10000 nM T12091 C5VPH9 16129448 IC50 > 10000 nM T12091 CPQ31L 25195294 IC50 = 17 nM T12091 CN2QG1 44223357 IC50 = 33.3 nM T12091 C3VRO9 44557921 IC50 > 10000 nM T12091 CXO0M2 46173038 IC50 = 35 nM T12091 CDV74N 50997747 IC50 = 107.9 nM T12091 C91FTP 57339386 IC50 = 110 nM T12091 CIP7B1 60182373 IC50 = 43 nM T12091 CQ6KV9 60182388 IC50 = 26.2 nM T12091 C37NKO 67129970 IC50 > 10000 nM T12091 CK80LJ 67130050 IC50 > 10000 nM T12091 C8I7GC 68293638 IC50 > 10000 nM T12091 C7GRV2 68755406 IC50 > 10000 nM T12091 CZ5EL7 71299325 IC50 = 15 nM T12091 CZM1K4 71765510 IC50 = 7 nM T12091 CJ2T9E 76332983 IC50 = 220 nM T12091 C75CEZ 91933902 IC50 = 10 nM T12091 CYX7T2 117072549 IC50 = 5090 nM T12091 CY58WC 117603102 IC50 = 9 nM T12091 CARX34 118392555 IC50 = 17 nM T12091 CA4T2K 118392556 IC50 = 120 nM T12091 CJG8B0 118392559 IC50 = 790 nM T12091 C2ZP8O 118392562 IC50 = 63 nM T12091 C1FE4J 118392566 IC50 = 23 nM T12091 CSXJ76 118392567 IC50 = 110 nM T12091 CC6K3M 118392573 IC50 = 86 nM T12091 C3T8XG 118392586 IC50 = 10 nM T12091 CG2U0M 118664452 IC50 = 109 nM T12091 CCUF04 118664598 IC50 = 246 nM T12091 C4XV3S 118664606 IC50 = 291 nM T12091 C8OL9Q 118664623 IC50 = 19 nM T12091 CQ53IT 118664628 IC50 = 63 nM T12091 CR76HA 118664702 IC50 = 5990 nM T12091 C7B8FM 118664739 IC50 = 326 nM T12091 CN4OX8 118664795 IC50 = 47 nM T12091 C16PNO 118664834 IC50 = 1971 nM T12091 CS7RK6 118664846 IC50 = 422 nM T12091 CAM1Z6 118664858 IC50 = 29 nM T12091 CD4W1A 118664876 IC50 = 738 nM T12091 COJK75 118664883 IC50 = 796 nM T12091 C6E4TV 118664891 IC50 = 27 nM T12091 CP8SE9 118664894 IC50 = 48 nM T12091 CS7GM9 118664938 IC50 = 16 nM T12091 CXV5B6 118664997 IC50 = 1026 nM T12091 CA92ES 118665005 IC50 = 526 nM T12091 C69BRA 118665049 IC50 = 54 nM T12091 CKM5S6 118665074 IC50 = 93 nM T12091 C0YB8O 118665087 IC50 = 25 nM T12091 CDIY19 118716042 IC50 = 110 nM T12091 CTJ0Q7 118716043 IC50 = 270 nM T12091 C1DVT7 118716164 IC50 = 6 nM T12091 CPC0N1 118716165 IC50 = 14 nM T12091 CZD49P 118716166 IC50 = 1870 nM T12091 C87ZPY 118796358 IC50 = 5130 nM T12091 C2LD1B 121232401 IC50 = 1.2 nM T12091 CI2YE9 132606873 IC50 = 217 nM T12091 CA02UO 133107911 IC50 = 32 nM T12091 CALE74 134691232 IC50 = 13 nM T12091 CK6W9X 135567453 IC50 = 194 nM T12091 C6HU9E 135567454 IC50 = 42 nM T12091 CN8U0P 135908049 IC50 = 344 nM T12091 CFI59M 136315995 IC50 = 18200 nM T12091 C23NFG 136598555 IC50 = 8200 nM T12091 CI1E8V 137634241 IC50 > 10000 nM T12091 CPT0V7 138454752 IC50 = 9 nM T12091 COW4V7 139582022 IC50 = 5 nM T12091 CE28UJ 145982726 IC50 = 68 nM T12091 CTF13L 145982833 IC50 = 293 nM T12091 CTAU82 145982904 IC50 = 439 nM T12091 CQHR19 145983288 IC50 = 2300 nM T12091 CTQ6X1 145983297 IC50 = 220 nM T12091 C6CV2P 145983361 IC50 = 1525 nM T12091 CNS8G0 145983444 IC50 = 165 nM T12091 C61BLQ 145983489 IC50 = 1000 nM T12091 CO89IY 145983541 IC50 = 138 nM T12091 CC09YN 145983872 IC50 = 186 nM T12091 C0YAQ3 145983889 IC50 = 653 nM T12091 C14KEW 145985284 IC50 = 167 nM T12091 CR6S8Z 145985704 IC50 = 431 nM T12091 CDB91R 145985727 IC50 = 10 nM T12091 C8ND3A 145985792 IC50 = 248 nM T12091 CUJ6Z5 145985892 IC50 = 91 nM T12091 CG1B7D 145986044 IC50 = 383 nM T12091 CBJ5N9 145986265 IC50 = 386 nM T12091 CT9UE5 155510654 IC50 < 2 nM T12091 CF2CU8 155510758 IC50 = 10 nM T12091 C1L9IF 155510984 IC50 < 2 nM T12091 CUA50Q 155512496 IC50 > 1000 nM T12091 C2MD1Q 155513187 IC50 > 10000 nM T12091 CQ64DF 155514482 IC50 = 7 nM T12091 CW6C2E 155514502 IC50 = 687 nM T12091 C5PA2F 155525040 IC50 = 712 nM T12091 C81AHZ 155525733 IC50 = 102 nM T12091 CJ71GR 155528153 IC50 > 1000 nM T12091 C9YMX3 155532969 IC50 = 5 nM T12091 CT23CQ 155544649 IC50 = 52 nM T12091 CL3V7C 155547885 IC50 = 694 nM T12091 CRY3A2 155548898 IC50 = 5 nM T12091 CUQ3O5 155548923 IC50 > 1000 nM T12091 C4T1BG 155550313 IC50 = 5 nM T12091 CY0A3R 155556360 IC50 = 751 nM T12091 C6UCG2 155562760 IC50 = 263 nM T12091 CWOE21 155564042 IC50 = 3 nM T12091 C31ECF 155564334 IC50 = 363 nM T12091 CK9Q5N 155564435 IC50 = 477 nM T12091 D05NEC 60182364 IC50 < 5 nM T12091 D06CMG 91754554 IC50 = 24 nM T12091 D0F2MP 60182389 IC50 < 5 nM T12091 D0PP6Y 60182393 IC50 = 53.4 nM T12091 D0RF7O 44577753 IC50 = 32 nM T12091 D0Y0BK 11524144 IC50 = 67.5 nM T60077 D02DGU 444795 Ki = 0.5 nM T60077 D0G3PI 449171 EC50 = 2.6 nM T60077 D0N0RU 82146 Ki = 5.9 nM T60077 D06QXI 9863342 EC50 = 2 nM T60077 D08JAC 5288209 Ki > 2800 nM T60077 D09DJC 9863341 EC50 = 0.8 nM T60077 D08GRF 5287705 Ki = 10.2 nM T60077 D09YUQ 127019 EC50 = 180 nM T60077 D0YO4D 3922 Ki = 7.5 nM T60077 CRI78W 94391 EC50 = 42000 nM T60077 CX90MS 128016 Ki = 640 nM T60077 C1E2FR 442048 EC50 = 32000 nM T60077 CZ8WQ4 584660 EC50 = 20000 nM T60077 CD3P5S 585022 EC50 = 35000 nM T60077 CXK08W 585035 EC50 = 48000 nM T60077 CZ7K5V 585049 EC50 = 8900 nM T60077 CT30JZ 585603 EC50 > 30000 nM T60077 C9JFT3 661071 EC50 = 8300 nM T60077 CMF7L1 737267 EC50 > 30000 nM T60077 CDVJ42 767163 EC50 > 30000 nM T60077 CWM95S 843040 EC50 = 16000 nM T60077 C5T2PS 843045 EC50 = 8800 nM T60077 CUHQ27 997606 EC50 = 29000 nM T60077 CZO04Y 1163179 IC50 = 11000 nM T60077 C30YVK 1169819 IC50 = 14000 nM T60077 C5UJF1 1637033 EC50 = 42000 nM T60077 CG3WZ4 2063265 EC50 > 30000 nM T60077 CG9DK0 2295706 IC50 = 12300 nM T60077 CSH2V8 2758079 EC50 = 13100 nM T60077 C4XZ0V 2758080 EC50 = 13000 nM T60077 CM60VP 2758604 EC50 = 18600 nM T60077 C1UT6Y 2758738 EC50 = 30000 nM T60077 C51INO 2886165 IC50 = 6000 nM T60077 CI8NO1 3025917 EC50 = 1600 nM T60077 C78QSL 3025918 EC50 = 300 nM T60077 CQ40OB 3025919 EC50 = 57 nM T60077 CYA2P5 3025934 EC50 = 3000 nM T60077 C0SBR8 3025935 EC50 = 2600 nM T60077 CK6X4W 3025936 EC50 = 1300 nM T60077 CK3N2G 3035780 EC50 = 980 nM T60077 CGL71X 6366726 EC50 = 23 nM T60077 CA5GS8 6438168 EC50 = 180 nM T60077 CGTB79 6440940 EC50 = 5200 nM T60077 CJHW10 6441985 IC50 > 1000 nM T60077 CVIT54 6491146 EC50 = 37000 nM T60077 CZ2N9P 7023630 EC50 = 28000 nM T60077 CG4FM8 7745122 EC50 = 370 nM T60077 CRXY80 7745146 EC50 = 310 nM T60077 C9SX8K 7745148 EC50 = 8600 nM T60077 CBE62R 9799320 EC50 = 100 nM T60077 COP9S7 9799477 EC50 = 3 nM T60077 CW7D0R 9810431 Ki = 191 nM T60077 CBV6Y2 9818688 EC50 = 1900 nM T60077 CEK1O4 9820039 EC50 = 210 nM T60077 CQFA96 9845057 Ki = 4 nM T60077 CQ1ZH6 9847065 Ki = 8.2 nM T60077 CAE0R3 9868664 Ki = 15.5 nM T60077 CRC51S 9869157 Ki = 5.2 nM T60077 CSK5B8 9885521 EC50 > 1000 nM T60077 C5AD1H 9886137 Ki = 8 nM T60077 CKNQ14 9887034 EC50 = 180 nM T60077 C90UXQ 9889347 Ki = 11.5 nM T60077 C8MK1Y 9889522 Ki = 400 nM T60077 C2WFX1 9905729 EC50 = 39 nM T60077 C0A3UZ 9911319 Ki = 3.9 nM T60077 C9VEF0 9949645 EC50 = 3200 nM T60077 C6JLI1 9973307 EC50 = 770 nM T60077 CVM8I3 9973559 EC50 = 6800 nM T60077 CAE52Z 9997909 EC50 = 1600 nM T60077 C7VS6O 9998151 EC50 = 33 nM T60077 CM1BQ5 10003577 Ki = 16 nM T60077 CZP71W 10022432 EC50 = 2000 nM T60077 C8RSG9 10043365 EC50 = 160 nM T60077 CC0N1S 10043729 EC50 = 33 nM T60077 CE60FI 10065757 Ki = 7 nM T60077 C2C0GJ 10066739 EC50 = 2300 nM T60077 CFQ1Y3 10073992 Ki = 10 nM T60077 C4VU6T 10087372 EC50 = 2400 nM T60077 CXL0Y3 10089642 EC50 = 1000 nM T60077 CC8R9M 10093918 Ki = 1200 nM T60077 C59GXP 10135960 Ki = 15 nM T60077 CO4S6H 10137005 EC50 = 157 nM T60077 CQYW32 10137940 Ki = 15 nM T60077 CP96OH 10204841 Ki = 4 nM T60077 CTKY45 10206438 Ki = 55 nM T60077 C90YNI 10207221 Ki = 12 nM T60077 C1O4PN 10207439 Ki = 10 nM T60077 C0AV2Z 10226478 Ki = 142 nM T60077 C0WRE7 10273807 Ki = 11 nM T60077 C6FT2B 10294841 EC50 = 37 nM T60077 C27ZPC 10297135 Ki = 261 nM T60077 CY1J5M 10308975 Ki = 4 nM T60077 C61TSO 10314077 EC50 = 2700 nM T60077 CUZR60 10314977 EC50 = 500 nM T60077 C6C5GP 10320109 Ki = 790 nM T60077 C2XBM9 10362613 EC50 = 47 nM T60077 CUEF37 10362997 IC50 = 50 nM T60077 CZTK13 10405638 EC50 = 500 nM T60077 CXA0N9 10458226 Ki = 1700 nM T60077 C0CHL5 10474101 EC50 = 140 nM T60077 CL31KB 10499086 EC50 = 207 nM T60077 CF87BZ 10523774 EC50 = 377 nM T60077 C2TP9D 10598286 Ki = 623 nM T60077 CS96IV 10619935 EC50 = 9 nM T60077 C4TO6H 10620598 EC50 = 12 nM T60077 CE1OC7 10644298 Ki > 1000 nM T60077 CH3D5N 10645862 Ki > 1000 nM T60077 CVQ6L1 10759115 EC50 = 3700 nM T60077 C8UG3F 10926235 EC50 = 25 nM T60077 CC40ME 11793226 Ki = 120 nM T60077 C0WA5F 11793407 Ki = 2 nM T60077 C4QYX8 11962184 Ki = 12 nM T60077 C38KZG 11978565 EC50 = 87000 nM T60077 C1AOP8 11978570 EC50 = 20000 nM T60077 C5TS1Q 13413729 EC50 = 5500 nM T60077 CJ74NB 16794302 EC50 > 30000 nM T60077 C3P6XD 19002087 EC50 = 130 nM T60077 CVA8T2 20117108 IC50 = 22400 nM T60077 CY7P2M 20707149 EC50 = 61 nM T60077 CV1C4A 22226112 EC50 > 1000 nM T60077 C41JDY 22400850 EC50 > 30000 nM T60077 CA59NU 22686157 EC50 > 30000 nM T60077 C0M9JB 22688013 EC50 = 18000 nM T60077 CP2CA5 23005221 EC50 = 150 nM T60077 C15NSJ 24828803 EC50 = 10300 nM T60077 CO31MA 24828805 EC50 = 7800 nM T60077 CW51RK 24828806 EC50 = 3100 nM T60077 C9N4PO 25195030 IC50 = 870 nM T60077 CQUB90 25195031 IC50 = 750 nM T60077 C0A2XU 29288275 EC50 = 2100 nM T60077 CT4J7Z 41500207 IC50 = 10900 nM T60077 CPA87R 44287651 Ki = 12 nM T60077 C1K8FB 44287715 Ki = 64.5 nM T60077 CI83JY 44287875 Ki = 33 nM T60077 CH8T3V 44325132 EC50 = 180 nM T60077 C1KUN0 44325759 Ki = 124 nM T60077 CLB6X7 44325767 Ki > 1000 nM T60077 CW0T6K 44353336 Ki = 3.9 nM T60077 C8K0AB 44353347 Ki = 24.4 nM T60077 C3DYE9 44353422 Ki = 7.4 nM T60077 C5DTY3 44353441 Ki = 2.4 nM T60077 C2M8TN 44353456 Ki = 9.9 nM T60077 CVKA40 44353466 Ki = 12.3 nM T60077 C8J5SA 44353480 Ki = 17.2 nM T60077 CIB15X 44353481 Ki = 8.5 nM T60077 C1AM4Y 44377164 Ki > 1000 nM T60077 C05RAC 44377446 Ki = 14 nM T60077 CPW0M2 44377447 Ki = 91 nM T60077 CDU3F0 44410404 Ki = 161 nM T60077 CRW3F9 44410405 EC50 = 169 nM T60077 CJX92G 44410453 Ki = 63 nM T60077 C1YKC7 44410518 Ki = 188 nM T60077 CI64YQ 44410534 EC50 = 151 nM T60077 CCS4X0 44410540 Ki = 88 nM T60077 CQVY89 44410541 Ki = 24 nM T60077 CLR9U4 44410562 Ki = 126 nM T60077 CXI98E 44410565 EC50 = 52 nM T60077 C0ZIF2 44410568 EC50 = 216 nM T60077 CW4YU7 44410575 Ki = 34 nM T60077 CV0TB9 44410576 Ki = 238 nM T60077 C9L6TA 44410610 EC50 = 98 nM T60077 CKY50J 44410620 EC50 = 117 nM T60077 CO2AF5 44410623 Ki = 72 nM T60077 C2R7KB 44410653 Ki = 327 nM T60077 C2QW1R 44410654 Ki = 185 nM T60077 CRI0J3 44460654 Ki > 2800 nM T60077 CEA20Z 44571531 IC50 > 10000 nM T60077 CG02HN 44571532 IC50 > 10000 nM T60077 CDZ84V 44571568 IC50 = 3000 nM T60077 CF21WB 44571569 IC50 = 3900 nM T60077 CA9FT0 44571643 IC50 > 10000 nM T60077 C5ZX4B 54597874 IC50 > 10000 nM T60077 CB84WZ 59205486 EC50 = 12800 nM T60077 CIO69D 59853119 EC50 = 16200 nM T60077 CNR48W 62216411 EC50 > 30000 nM T60077 C9S5EN 64222254 EC50 = 21000 nM T60077 CX1P8I 67042254 IC50 > 10000 nM T60077 CGL2E4 70868689 EC50 = 6700 nM T60077 CCX30R 71717207 Ki > 2800 nM T60077 CVW1H0 73350281 Ki = 12 nM T60077 CBG04C 80198302 EC50 = 13400 nM T60077 C3PI7Z 82483008 EC50 = 6600 nM T60077 C2WG9L 138393074 EC50 = 4500 nM T60077 C2OJ9E 141259219 EC50 = 11700 nM T60077 C7N6KH 145950441 EC50 = 13900 nM T60077 CRTB69 145952096 EC50 = 2200 nM T60077 CLND09 145957286 EC50 = 27100 nM T60077 CO5LP2 145959006 EC50 = 16000 nM T60077 CM8T6X 145982686 EC50 = 16000 nM T60077 C1QZ7W 145986715 IC50 = 18000 nM T60077 C7X3AL 153763221 EC50 = 6000 nM T60077 CUNF95 155513665 EC50 = 22300 nM T60077 C3Z6VL 155514089 EC50 = 11100 nM T60077 CGO6X4 155515480 EC50 = 4300 nM T60077 CWR01U 155517898 EC50 > 30000 nM T60077 C7DN5A 155520617 EC50 > 30000 nM T60077 CT4HM2 155524204 EC50 = 7000 nM T60077 C95KYP 155526365 EC50 = 3800 nM T60077 C2QTX3 155530866 EC50 = 2100 nM T60077 C4JD0I 155531001 EC50 = 9900 nM T60077 CE7I8Q 155534885 EC50 = 43000 nM T60077 CX2JR0 155535627 EC50 = 3100 nM T60077 CE7OD6 155538138 EC50 = 290 nM T60077 C1TMV9 155539075 EC50 = 1900 nM T60077 CEM97Q 155539095 EC50 = 10000 nM T60077 C7E9KD 155539294 EC50 = 5300 nM T60077 CK02XE 155539921 EC50 = 6600 nM T60077 CR9Y8W 155541027 EC50 = 8900 nM T60077 CP3I4H 155541634 EC50 = 1400 nM T60077 C2QGR5 155549327 EC50 = 10100 nM T60077 C80ZVT 155556139 EC50 > 30000 nM T60077 CIO4S2 155557691 EC50 = 143 nM T60077 CM52UW 155560868 EC50 = 2300 nM T60077 CG3D8J 155564760 EC50 = 800 nM T60077 CX7OR2 155566024 EC50 = 12000 nM T60077 D02YHD 11755040 IC50 = 44 nM T60077 D09XCX 5694 EC50 = 13000 nM T60077 D0G6JM 5289501 EC50 > 10000 nM T60077 D0Q9FZ 6442223 Ki = 9 nM T63393 CHDJ89 53358775 IC50 > 30000 nM T63393 C37KDG 53358900 IC50 > 30000 nM T63393 C7GTQ9 71449523 IC50 > 20000 nM T63393 CA1CL3 71451318 IC50 > 30000 nM T63393 CC4D7M 71456641 IC50 = 5000 nM T63393 CAVM60 71460332 IC50 = 2000 nM T63393 C2JS8B 71462027 IC50 = 7000 nM T63393 D02FGK 53358901 IC50 > 30000 nM T97747 D0NR6S 3002977 IC50 = 1.3 nM T97747 D00XBC 46861584 IC50 = 6309.57 nM T97747 D09JLI 3009355 IC50 = 1.2 nM T97747 D0F7PZ 53316710 IC50 < 0.1 nM T97747 D0O2XQ 11256587 IC50 > 10000 nM T97747 D0O9UC 5275766 IC50 = 3.5 nM T97747 D0Y7NA 49871007 IC50 = 3.1 nM T97747 D0YQ7U 11285792 IC50 = 3 nM T97747 D07GIB 11614352 IC50 = 0.26 nM T97747 D0G6JE 9574343 Ki = 2.1 nM T97747 D0G6SZ 3001322 IC50 = 5.623 nM T97747 D0Q2JS 10436045 Ki = 4260 nM T97747 D0W0LS 183789 IC50 = 1.2 nM T97747 C7Y8VS 1318 EC50 = 4900 nM T97747 CB4Z9P 1474 EC50 = 19000 nM T97747 C78GSK 14338 EC50 = 11000 nM T97747 CW6J7R 15664 EC50 = 2300 nM T97747 CBX47E 20445 IC50 = 501187.23 nM T97747 CD72TB 65237 EC50 = 63095.73 nM T97747 CF1UA4 70848 IC50 = 25000 nM T97747 CR15FN 72791 EC50 > 1000000 nM T97747 C8SC9N 72792 EC50 = 2511.89 nM T97747 C7SIE4 74265 EC50 = 1000 nM T97747 CMJ4V7 77524 EC50 < 1000000 nM T97747 CGZ1C6 77865 EC50 < 1000000 nM T97747 CBW4N5 93149 EC50 = 1800 nM T97747 CTUE81 336912 IC50 = 587000 nM T97747 C2P3FM 353741 IC50 = 199526.23 nM T97747 CW39FG 455656 Ki = 31 nM T97747 C91RPQ 455657 Ki = 32 nM T97747 CLU42H 456292 Ki = 18 nM T97747 CJKB92 456293 Ki = 28 nM T97747 C2K7SR 456298 Ki = 62 nM T97747 CG48QX 456319 IC50 = 90 nM T97747 CN37SU 456323 Ki = 5 nM T97747 C9RGE7 456339 Ki = 15 nM T97747 C70ZGM 456372 Ki = 5 nM T97747 CSOT95 456374 IC50 = 255 nM T97747 CDCZ30 456375 Ki = 1 nM T97747 C4AW8L 456611 Ki = 44 nM T97747 C2VJ3Z 456615 IC50 = 440 nM T97747 CC02UF 456647 Ki = 30 nM T97747 CP3R6C 457671 Ki = 54 nM T97747 CPK6B5 457672 Ki = 29 nM T97747 CNU94V 457679 IC50 = 200 nM T97747 CH6J1S 457797 IC50 > 1000 nM T97747 C42WYA 457829 IC50 > 1000 nM T97747 C9D5BT 457845 IC50 = 980 nM T97747 C78ICG 457871 IC50 = 0.5 nM T97747 C43TRB 457874 Ki = 11 nM T97747 CTU5D6 457875 Ki = 58 nM T97747 C2FHD7 461327 Ki = 5 nM T97747 C8FQ6Y 461546 Ki = 440 nM T97747 CUWT43 461838 Ki = 230 nM T97747 C38ERL 461871 Ki = 45 nM T97747 CHG02J 462395 Ki = 2.7 nM T97747 CR64WQ 462409 Ki = 7 nM T97747 CU43EI 462571 Ki = 10 nM T97747 C47MIH 462573 Ki = 5.23 nM T97747 CKI1S3 462772 Ki = 49 nM T97747 C9YW6M 462902 Ki = 20 nM T97747 CCHZ81 462989 Ki = 18 nM T97747 CF8X4A 463209 Ki = 11 nM T97747 CNVX67 463210 Ki = 11 nM T97747 C2HB4T 463319 Ki = 12 nM T97747 CC85IE 463493 Ki > 1300 nM T97747 C2T0PC 463502 Ki = 74 nM T97747 CH61SC 463517 Ki = 442 nM T97747 C8UQ6H 463616 Ki = 0.7 nM T97747 CVQ5L9 463892 Ki = 11 nM T97747 CAP7I1 464036 Ki = 2 nM T97747 CU29RH 471179 IC50 = 35 nM T97747 C2P0CD 473081 IC50 = 480 nM T97747 C0P7LR 473305 IC50 = 152 nM T97747 CTB56C 474188 Ki = 38 nM T97747 CZ49VF 474465 Ki = 352 nM T97747 CSF9B6 478296 IC50 = 35 nM T97747 CWC96R 478302 IC50 = 30 nM T97747 CRW43A 478307 IC50 = 30 nM T97747 CRF63Q 478308 IC50 = 120 nM T97747 CTF02S 478387 IC50 = 60 nM T97747 C4CD1U 478399 IC50 = 260 nM T97747 C7MVA1 478409 IC50 = 200 nM T97747 CZFM52 478410 IC50 = 25 nM T97747 C2XZ0N 478412 IC50 = 70 nM T97747 CS1NU8 478413 IC50 = 650.13 nM T97747 CTK7B5 478414 IC50 = 50 nM T97747 C0HPV2 478418 IC50 = 120.23 nM T97747 C40OJQ 478439 IC50 = 120.23 nM T97747 C9RM0U 478440 IC50 = 100 nM T97747 C84EFC 478444 IC50 = 4 nM T97747 C6DU8Z 478445 IC50 = 2.5 nM T97747 C79FCT 478446 IC50 = 6 nM T97747 C7BKL5 478447 IC50 = 75 nM T97747 CP60TK 478448 IC50 = 20 nM T97747 CA90RU 478449 IC50 = 100 nM T97747 CC91KL 478450 IC50 = 3.02 nM T97747 C67UKD 478451 IC50 = 3.981 nM T97747 C35VTN 478452 IC50 = 19.95 nM T97747 CF43WD 478471 IC50 > 10000 nM T97747 C1G8DT 478475 IC50 > 10000 nM T97747 CL2CY9 478493 IC50 = 340 nM T97747 CD7NT2 478494 IC50 = 850 nM T97747 CV82HX 478495 IC50 = 1400 nM T97747 CX6WB9 478496 IC50 = 100 nM T97747 C76GKH 478499 IC50 = 70 nM T97747 CP67RF 478500 IC50 = 40 nM T97747 CJ0M6N 478501 IC50 = 150 nM T97747 C0R4CK 478502 IC50 = 60 nM T97747 CH1P4S 478503 IC50 = 40 nM T97747 CPXW62 478508 IC50 > 4000 nM T97747 C2N0BX 478512 IC50 = 340 nM T97747 C10YWE 479835 IC50 = 450 nM T97747 C7TG2M 479837 IC50 = 2000 nM T97747 C2TSP5 479838 IC50 = 1300 nM T97747 CHK75U 479846 IC50 = 90 nM T97747 CE57HZ 479847 IC50 = 110 nM T97747 CQW7Z2 479852 IC50 = 180 nM T97747 CEWR08 479853 IC50 = 110 nM T97747 CW79PV 479855 IC50 > 1000 nM T97747 C8IQ7L 479856 IC50 > 1000 nM T97747 CCHZ69 479857 IC50 = 3000 nM T97747 CR8TC2 479858 IC50 = 100 nM T97747 CVO0B9 479859 IC50 = 110 nM T97747 CT3V4Z 479860 IC50 = 500 nM T97747 CDPW28 479861 IC50 > 1000 nM T97747 C89LZS 479863 IC50 ~ 10000 nM T97747 CR1F7T 479864 IC50 ~ 1000 nM T97747 C0W1KP 479865 IC50 = 200 nM T97747 CEUX01 479866 IC50 > 1000 nM T97747 CBY3Z7 479867 IC50 = 300 nM T97747 C8IMJ5 479868 IC50 = 160 nM T97747 CJ6R0N 479870 IC50 = 570 nM T97747 C8GE2D 479871 IC50 = 60 nM T97747 CKI69Y 479872 IC50 = 180 nM T97747 CX5T0U 479873 IC50 = 110 nM T97747 CAX24K 479874 IC50 > 1000 nM T97747 CCF3N1 479876 IC50 = 400 nM T97747 CJC18Q 479877 IC50 = 100 nM T97747 C6R8FZ 479878 IC50 ~ 10000 nM T97747 C5WRD1 479879 IC50 > 10000 nM T97747 C6OQ5C 479883 IC50 = 80 nM T97747 CT78SG 482147 IC50 = 100 nM T97747 CMZ6P3 482148 IC50 = 50 nM T97747 C35QRN 482150 IC50 = 300 nM T97747 COIA12 482217 IC50 ~ 10000 nM T97747 CKIZ45 483330 IC50 = 15 nM T97747 C6XI2W 483331 IC50 = 27 nM T97747 C4YDE0 483332 IC50 = 111 nM T97747 CCN9V1 483333 IC50 = 335 nM T97747 CAE58G 483334 IC50 = 23 nM T97747 CKU10W 483335 IC50 = 15 nM T97747 C57XVT 483336 IC50 = 15 nM T97747 CN5F7J 483337 IC50 = 16 nM T97747 C7K9DZ 483338 IC50 = 28 nM T97747 CQ3KO7 483339 IC50 = 25 nM T97747 C7AP9W 483340 IC50 = 4 nM T97747 CAB79M 483341 IC50 = 246 nM T97747 C7XW2D 483342 IC50 = 48 nM T97747 C7PMT6 483343 IC50 = 112 nM T97747 CP25RI 483344 IC50 = 10 nM T97747 C9XV0W 483345 IC50 = 18 nM T97747 CDXH14 483348 IC50 = 8600 nM T97747 C6XJ4V 483350 IC50 = 88000 nM T97747 C39BFX 483351 IC50 = 7200 nM T97747 C1T3LZ 483352 IC50 = 24000 nM T97747 CE71IM 483353 IC50 = 4400 nM T97747 C9SUH2 483354 IC50 = 6800 nM T97747 C17BMC 483355 IC50 = 3800 nM T97747 CY7TI4 483356 IC50 = 11000 nM T97747 C1NGQ0 483360 IC50 = 15000 nM T97747 C78PDK 483361 IC50 = 2300 nM T97747 C1FAV4 483362 IC50 = 10400 nM T97747 CI01WP 483363 IC50 = 3500 nM T97747 CH3AK8 483364 IC50 = 8400 nM T97747 CVQG07 483369 IC50 = 1.5 nM T97747 C9SAP8 483382 IC50 = 2 nM T97747 C6EP7Q 483407 EC50 = 1 nM T97747 CN2M0Z 483741 Ki = 590 nM T97747 CTO42Z 483744 Ki = 20 nM T97747 C1TRZ6 483746 Ki = 1300 nM T97747 C4J8NF 483747 IC50 = 0.01 nM T97747 C6E4JZ 484577 Ki = 5 nM T97747 CBLP57 484578 Ki = 3 nM T97747 CQX89C 484579 Ki = 5 nM T97747 C2PZO7 484581 Ki = 8 nM T97747 CAXL81 486595 IC50 = 400 nM T97747 C8KY2N 486601 IC50 = 2 nM T97747 CC17IT 486602 IC50 = 4 nM T97747 CUJ4P3 486604 IC50 = 1.5 nM T97747 C1F4ZP 486605 IC50 = 0.8 nM T97747 C7UVY2 486606 IC50 = 2 nM T97747 CTG0K5 486607 IC50 = 3 nM T97747 C0N1KQ 486608 IC50 = 120 nM T97747 CT8JO0 486632 IC50 = 1.5 nM T97747 CP6ZN1 489305 IC50 = 6.5 nM T97747 C64KTB 489306 IC50 = 3 nM T97747 C97FKT 489307 IC50 = 4 nM T97747 C6EAD2 489308 IC50 = 2 nM T97747 CD9CA1 489312 IC50 = 25 nM T97747 C0GS3N 489313 IC50 = 41 nM T97747 CL5UD4 489314 IC50 = 60 nM T97747 CHUB62 489315 IC50 = 0.3 nM T97747 C90YRJ 489316 IC50 = 6.5 nM T97747 C91OWI 489593 IC50 > 10000 nM T97747 C7QDT0 489594 IC50 = 26 nM T97747 C9Q8MV 489595 IC50 = 49 nM T97747 CFZ02X 489596 IC50 > 10000 nM T97747 CP15BS 489597 IC50 = 3500 nM T97747 CZ39NR 489598 IC50 > 10000 nM T97747 CWM08J 489599 IC50 > 10000 nM T97747 C6AD2R 489805 IC50 = 610 nM T97747 CLB6T9 489806 IC50 = 67 nM T97747 C03VWO 489807 IC50 = 155 nM T97747 CVR7Q0 489808 IC50 = 52 nM T97747 C4HO2V 489809 IC50 = 94 nM T97747 CBO93F 489810 IC50 = 750 nM T97747 CRXG81 489811 IC50 = 140 nM T97747 CO7AN1 489812 IC50 = 140 nM T97747 CLU42C 489813 IC50 > 1000 nM T97747 C6BLV4 489814 IC50 = 97 nM T97747 C7XR9V 489815 IC50 = 96 nM T97747 C04MOK 489816 IC50 = 89 nM T97747 C38MNQ 489817 IC50 = 48 nM T97747 CWP0O9 489818 IC50 = 32 nM T97747 CBGQ95 489820 IC50 = 260 nM T97747 CR78CU 489821 IC50 = 55 nM T97747 CS3Q6D 489822 IC50 = 46 nM T97747 CM78TR 489823 IC50 = 33 nM T97747 CK25FT 489824 IC50 = 34 nM T97747 CXV7H5 489825 IC50 = 19 nM T97747 CJQF51 489826 IC50 = 48 nM T97747 CLB51I 489827 IC50 = 57 nM T97747 C4WES0 489828 IC50 > 1000 nM T97747 CNU5F6 489829 IC50 = 810 nM T97747 C20OGE 489830 IC50 > 1000 nM T97747 C6L0XZ 489831 IC50 > 1000 nM T97747 CG24QV 489832 IC50 > 1000 nM T97747 CE09IT 489833 IC50 = 390 nM T97747 CYA56U 489834 IC50 > 1000 nM T97747 C9K7VD 489835 IC50 = 150 nM T97747 CA4KS9 490006 IC50 = 46 nM T97747 CIYP51 490007 IC50 = 31 nM T97747 C8OH9Y 490008 IC50 = 12 nM T97747 C8MH9R 490010 IC50 = 17 nM T97747 C1ZY4G 490011 IC50 = 15 nM T97747 C7QR3K 490012 IC50 = 9 nM T97747 C7PF8H 490013 IC50 = 5 nM T97747 CBG64R 490014 IC50 = 2 nM T97747 CQZW31 490016 IC50 = 4 nM T97747 C15GOK 490017 IC50 = 2 nM T97747 CV06XI 490018 IC50 = 0.1 nM T97747 C9YNU2 490019 IC50 = 0.2 nM T97747 CP8MR9 490020 IC50 = 0.8 nM T97747 C4R0QW 490022 IC50 = 0.8 nM T97747 C3PH6B 490023 IC50 = 0.2 nM T97747 CA5BZ8 491773 IC50 = 38 nM T97747 C9NE3B 496970 IC50 = 100 nM T97747 CI7GR8 496971 IC50 = 3 nM T97747 CJVQ67 496972 IC50 = 10 nM T97747 CQKL02 496973 IC50 = 5.998 nM T97747 CZ0W8A 496974 IC50 = 5 nM T97747 C6EDZ1 496975 IC50 = 2 nM T97747 C5BP9E 496983 IC50 = 6.998 nM T97747 CZ67QC 496984 IC50 = 5.998 nM T97747 CN9OE4 496985 IC50 = 12 nM T97747 C5HGF3 501043 IC50 = 1 nM T97747 CU4R2W 501044 IC50 = 3.6 nM T97747 C1GA2L 501045 IC50 = 1 nM T97747 CQ38YL 501046 IC50 = 0.5 nM T97747 C7TYW3 501047 IC50 = 1 nM T97747 C0YM7T 501048 IC50 = 24 nM T97747 C3GTE7 501049 IC50 = 4 nM T97747 CSYH30 501050 IC50 = 5 nM T97747 C2XT8B 501051 IC50 = 0.7998 nM T97747 CUR04D 501052 IC50 = 2 nM T97747 CGD5I0 501053 IC50 = 3 nM T97747 C6YVK3 501054 IC50 = 5.998 nM T97747 CZYS12 501055 IC50 = 0.1 nM T97747 C0L6BS 501056 IC50 = 0.7 nM T97747 CR3K8B 501057 IC50 = 3.999 nM T97747 C4R8TH 501058 IC50 = 36 nM T97747 CWL94S 501059 IC50 = 3 nM T97747 C4EYK5 501060 IC50 = 0.1 nM T97747 CP8ON7 501062 IC50 = 0.1 nM T97747 C0Y7TL 501063 IC50 = 0.2 nM T97747 C7JQ2Z 502259 Ki = 10 nM T97747 C9N6LP 503637 Ki = 5.1 nM T97747 CN7P0G 505865 IC50 = 300 nM T97747 CSAM47 505866 IC50 = 9 nM T97747 C40MHP 505867 IC50 = 10 nM T97747 C3WXP0 505868 IC50 = 12 nM T97747 CF8TK4 505869 IC50 = 6 nM T97747 CZ0KC5 505870 IC50 = 9 nM T97747 C2A1QX 505873 IC50 = 12 nM T97747 C15FCB 505874 IC50 = 66 nM T97747 C43SIR 505875 IC50 = 12 nM T97747 CQ9S3K 505876 IC50 = 42 nM T97747 CSZ3V1 505878 IC50 = 3.9 nM T97747 CJ24LQ 505879 IC50 = 5 nM T97747 CSIQ81 505880 IC50 = 6.6 nM T97747 CJ4P1O 505881 IC50 = 1.6 nM T97747 CD09FO 511294 Ki = 68 nM T97747 CZHY61 511295 Ki = 110 nM T97747 CC0WK3 511296 Ki = 86 nM T97747 C2YCQ4 511297 Ki = 360 nM T97747 CS61JO 511298 Ki = 190 nM T97747 CQE5N9 511299 Ki = 62 nM T97747 CN25FS 511303 Ki = 33 nM T97747 COCZ64 511304 Ki = 25 nM T97747 C2Z4CB 511305 Ki = 55 nM T97747 CU5DY2 511306 Ki = 155 nM T97747 CPW6C4 511307 Ki = 33 nM T97747 CC70RW 511308 Ki = 596 nM T97747 C1YFM7 511309 Ki = 8 nM T97747 CFJ63U 511332 Ki = 7 nM T97747 C49UTP 516172 IC50 = 1.199 nM T97747 CFY12E 516173 IC50 = 1.5 nM T97747 C17QUG 516174 IC50 = 2.3 nM T97747 CE7IZ3 516175 IC50 = 1.1 nM T97747 CAK7I5 516176 IC50 = 1.3 nM T97747 CJKA08 516177 IC50 = 2.2 nM T97747 CJ10ZD 516178 IC50 = 1.1 nM T97747 CLNW94 516179 IC50 = 2.6 nM T97747 C36DAX 516180 IC50 = 5 nM T97747 C17OWX 516181 IC50 = 1.3 nM T97747 CTR8J0 516182 IC50 = 2 nM T97747 CIT5M7 516183 IC50 = 3.2 nM T97747 CWI3S4 516184 IC50 = 3.1 nM T97747 C9H8KU 516185 IC50 = 1.7 nM T97747 C5XTV2 516186 IC50 = 3.5 nM T97747 C8AEM1 516187 IC50 = 1.3 nM T97747 CPE45H 516188 IC50 = 13.1 nM T97747 CF2ER3 516189 IC50 = 1.3 nM T97747 CZDN60 516190 IC50 = 1 nM T97747 C19ZRH 516191 IC50 = 0.8 nM T97747 C3VUY8 516192 IC50 = 0.5 nM T97747 C2UA5G 516193 IC50 = 1 nM T97747 C68PSM 516194 IC50 = 0.6 nM T97747 C2U3FJ 516195 IC50 = 0.8 nM T97747 C8T4PC 516196 IC50 = 0.6 nM T97747 C02BWL 516197 IC50 = 0.8 nM T97747 CA3W8V 516198 IC50 = 0.5 nM T97747 CICH26 516199 IC50 = 0.6 nM T97747 CQ1PG6 516200 IC50 = 0.8 nM T97747 CKI1J9 516201 IC50 = 0.4 nM T97747 CUX94K 516202 IC50 = 0.3 nM T97747 CNCR59 516203 IC50 = 0.9 nM T97747 C3A9RP 516204 IC50 = 1.2 nM T97747 CN80KP 516205 IC50 = 0.5 nM T97747 CTAR48 516206 IC50 = 2.1 nM T97747 C4Y1EX 516207 IC50 = 1.3 nM T97747 CMH39L 516208 IC50 = 0.9 nM T97747 CXD32U 516209 IC50 = 0.6 nM T97747 CB0PW1 516211 IC50 = 1.2 nM T97747 C9MVL1 516212 IC50 = 0.6 nM T97747 C2ISE5 516213 IC50 = 0.9 nM T97747 CBEO51 516214 IC50 = 1.1 nM T97747 CR15ZC 516215 IC50 = 1 nM T97747 CNSQ90 516216 IC50 = 0.3 nM T97747 CJUT37 516217 IC50 = 1.3 nM T97747 CMZ6C3 516218 IC50 = 0.8 nM T97747 C1F7HO 516219 IC50 = 1.3 nM T97747 C7SLM0 516220 IC50 = 0.7 nM T97747 CRD07L 516221 IC50 = 0.4 nM T97747 C97TAX 516222 IC50 = 1.1 nM T97747 CRG4W0 516223 IC50 = 0.6 nM T97747 C4BX1V 516224 IC50 = 0.3 nM T97747 CE1DA2 516225 IC50 = 1.4 nM T97747 C2WHI5 516226 IC50 = 1.5 nM T97747 CJ7E9S 516227 IC50 = 0.5 nM T97747 C23VSR 516228 IC50 = 0.5 nM T97747 C70EVZ 516229 IC50 = 0.7 nM T97747 CC8HS5 516230 IC50 = 0.4 nM T97747 CJ02LM 516231 IC50 = 0.3 nM T97747 CK1U5W 516232 IC50 = 0.3 nM T97747 C9UOI0 516233 IC50 = 0.3 nM T97747 C5D1XY 516234 IC50 = 0.3 nM T97747 C67BKT 516235 IC50 = 0.3 nM T97747 CL2KZ5 516236 IC50 = 0.9 nM T97747 CW9M7J 516237 IC50 = 0.5 nM T97747 CDTJ57 516238 IC50 = 1.6 nM T97747 CWTN29 516239 IC50 = 1.3 nM T97747 C0CAK2 516240 IC50 = 1.1 nM T97747 CV6JB5 516241 IC50 = 2.7 nM T97747 C4MG1X 516242 IC50 = 0.8 nM T97747 CGT3M2 516243 IC50 = 1.2 nM T97747 CM4D9P 516244 IC50 = 0.8 nM T97747 C4HF7G 516245 IC50 = 0.3 nM T97747 C6L1BX 516246 IC50 = 0.4 nM T97747 C4MQR0 516247 IC50 = 1.6 nM T97747 CK64CJ 516248 IC50 = 0.5 nM T97747 C1MP9U 516249 IC50 = 0.5 nM T97747 CA0CL5 516250 IC50 = 0.6 nM T97747 CIOG73 516251 IC50 = 0.5 nM T97747 CHZ03N 516252 IC50 = 0.6 nM T97747 CSWV89 516253 IC50 = 0.6 nM T97747 C1LB4X 516254 IC50 = 2.6 nM T97747 CA02XT 516255 IC50 = 0.4 nM T97747 CI76WJ 516256 IC50 = 0.2 nM T97747 C8SLJ6 516257 IC50 = 0.2 nM T97747 C5JO7X 516258 IC50 = 0.8 nM T97747 C1ZBU6 516259 IC50 = 0.5 nM T97747 CQ52IA 516260 IC50 = 0.7998 nM T97747 CJ71SM 516261 IC50 = 1.1 nM T97747 CDSF01 516262 IC50 = 0.3 nM T97747 CBEN83 516263 IC50 = 2.3 nM T97747 C65AZI 516264 IC50 = 1.3 nM T97747 CVK8R9 516266 IC50 = 1.6 nM T97747 C4Z1UM 516267 IC50 = 1.1 nM T97747 CCD9S6 516268 IC50 = 1.5 nM T97747 C72UXL 516269 IC50 = 0.7 nM T97747 CMJZ98 516270 IC50 = 0.9 nM T97747 C3ORY7 516271 IC50 = 0.4 nM T97747 CUB96H 516272 IC50 = 0.8 nM T97747 C86FJD 516273 IC50 = 0.8 nM T97747 C8JI6P 516274 IC50 = 0.4 nM T97747 COA04U 516275 IC50 = 0.7 nM T97747 C59YWP 516276 IC50 = 0.7 nM T97747 C75MOZ 516277 IC50 = 2 nM T97747 CIJX71 516278 IC50 = 1.1 nM T97747 C8ZT2N 516279 IC50 = 0.4 nM T97747 C9XU6R 516280 IC50 = 0.6 nM T97747 CSU21I 516281 IC50 = 0.6 nM T97747 CA56QB 516282 IC50 = 0.5 nM T97747 C28OFN 516283 IC50 = 1.1 nM T97747 CHN28A 516284 IC50 = 1.2 nM T97747 C8DAC7 516285 IC50 = 0.7 nM T97747 C5L4MQ 516286 IC50 = 0.9 nM T97747 CJ8NY1 516287 IC50 = 0.7 nM T97747 CY1B6X 516288 IC50 = 0.2 nM T97747 C1I4UL 516289 IC50 = 0.2 nM T97747 CK93QH 516290 IC50 = 0.6 nM T97747 CFKI94 516291 IC50 = 0.6 nM T97747 CBYO78 516292 IC50 = 0.4 nM T97747 C4XN2D 516293 IC50 = 0.6 nM T97747 C9D5QE 516294 IC50 = 1.6 nM T97747 CN8XA2 516295 IC50 = 1.1 nM T97747 CK1PD5 516296 IC50 = 1 nM T97747 CFEW91 516298 IC50 = 0.9 nM T97747 CDMW14 516299 IC50 = 1.5 nM T97747 C97KFD 516300 IC50 = 0.9 nM T97747 CBXT91 516301 IC50 = 1.5 nM T97747 CI5Q8L 516302 IC50 = 1.7 nM T97747 C8L2AF 516303 IC50 = 2.3 nM T97747 C8J2GI 516304 IC50 = 0.8 nM T97747 C2I3NA 516305 IC50 = 3.9 nM T97747 CN7MX3 516306 IC50 = 1.1 nM T97747 CZ23TX 516307 IC50 = 1 nM T97747 C6K0JX 516308 IC50 = 0.7 nM T97747 CL3P0C 516309 IC50 = 0.8 nM T97747 CV7JI2 516310 IC50 = 0.2 nM T97747 C81OXC 516311 IC50 = 0.5 nM T97747 C95XCF 516312 IC50 = 0.5 nM T97747 CNZ5I9 516313 IC50 = 0.5 nM T97747 CUAO78 516314 IC50 = 0.3 nM T97747 CG02IZ 516315 IC50 = 76 nM T97747 C1A0SH 516319 IC50 = 78 nM T97747 C92CLD 516325 IC50 = 2.198 nM T97747 C5Z9TB 516326 IC50 = 4.2 nM T97747 C3C0IU 516327 IC50 = 4.6 nM T97747 C0H9RE 516328 IC50 = 2.999 nM T97747 C8KPC3 516329 IC50 = 4.8 nM T97747 C3F0MY 516330 IC50 = 9 nM T97747 CUK2G8 516331 IC50 = 33 nM T97747 CGB36E 516332 IC50 = 2.999 nM T97747 CCJ4U8 516333 IC50 = 0.6 nM T97747 CAK2S5 516334 IC50 = 4.8 nM T97747 C8R5IX 516335 IC50 = 1.2 nM T97747 CK70CG 516336 IC50 = 1 nM T97747 CB14VJ 516337 IC50 = 0.6 nM T97747 COA15S 516338 IC50 = 20 nM T97747 CD8S9J 516339 IC50 = 2.3 nM T97747 C16UMB 516340 IC50 = 23 nM T97747 CQE9N8 516341 IC50 = 9 nM T97747 C7WHX0 516342 IC50 = 0.7998 nM T97747 C1EJM4 516343 IC50 = 1.199 nM T97747 CM1QB4 516344 IC50 = 22 nM T97747 CJ0BW8 516345 IC50 = 16 nM T97747 CZ54ST 516346 IC50 = 121.9 nM T97747 C8W3IM 516347 IC50 = 7.5 nM T97747 CDE5F0 516348 IC50 = 7.5 nM T97747 CF29PH 516349 IC50 = 16 nM T97747 C5DHL6 516350 IC50 = 9 nM T97747 CDAS93 516351 IC50 = 4 nM T97747 CH68TF 516352 IC50 = 12 nM T97747 CZ4YM1 516353 IC50 = 2.2 nM T97747 CAX3D4 516354 IC50 = 2.099 nM T97747 CCF0X5 516357 IC50 = 11.5 nM T97747 C1S2KP 516358 IC50 = 6.9 nM T97747 CE6O0T 516361 IC50 = 1.199 nM T97747 CKH2Z9 516362 IC50 = 1.199 nM T97747 CU32RP 516363 IC50 = 2.9 nM T97747 C3GA8B 516364 IC50 = 2.8 nM T97747 CE3FO7 516365 IC50 = 1.6 nM T97747 CNY7F9 516366 IC50 = 0.8995 nM T97747 C5R6OZ 516367 IC50 = 1.6 nM T97747 CJU93H 516368 IC50 = 5.5 nM T97747 CSF9D4 602123 IC50 = 125892.54 nM T97747 CXMY27 619353 IC50 = 501187.23 nM T97747 CYU56N 667748 IC50 = 8100 nM T97747 CMP4D3 1167892 EC50 = 3000 nM T97747 CAF8P7 2733927 EC50 = 19952.62 nM T97747 C90AHY 3002976 IC50 = 1 nM T97747 C1IPS0 3007227 IC50 = 105 nM T97747 CUY7J9 3008902 IC50 = 2 nM T97747 C1V4TU 3008903 IC50 = 80 nM T97747 CE3Q4V 3008904 IC50 = 2.8 nM T97747 CG7ZT5 3008905 IC50 = 3.8 nM T97747 C6VG7U 3008906 IC50 > 1000 nM T97747 C32FTI 3008907 IC50 = 100 nM T97747 CQR7S5 3008908 IC50 = 2 nM T97747 C8JLB6 3008909 IC50 = 27.3 nM T97747 C45FME 3008910 IC50 = 460 nM T97747 CC23PJ 3008911 IC50 = 102 nM T97747 CR3K2Z 3008912 IC50 = 43 nM T97747 CZ1V8Q 3008913 IC50 = 3 nM T97747 CDSG05 3008914 IC50 = 2.3 nM T97747 C4V0IN 3008915 IC50 > 1000 nM T97747 CKXR32 3008916 IC50 = 75 nM T97747 C1IS9G 3008917 IC50 = 0.7 nM T97747 CP12EY 3008918 IC50 = 7.8 nM T97747 CK83ZH 3008919 IC50 = 200 nM T97747 CEX1C8 3008920 IC50 > 100 nM T97747 CUNQ43 3008921 IC50 = 408 nM T97747 CI21SO 3008922 IC50 = 42 nM T97747 CU38DW 3008923 IC50 = 2.4 nM T97747 CI87PX 3008924 IC50 = 3.7 nM T97747 C2IW9S 3008925 IC50 = 31 nM T97747 C0PHV5 3008926 IC50 = 283 nM T97747 CZV0O6 3008927 IC50 = 1.1 nM T97747 C83ZWQ 3008928 IC50 = 1 nM T97747 CHQS14 3008929 IC50 = 3.3 nM T97747 C8KY7B 3008930 IC50 = 2.9 nM T97747 CH3L2R 3008931 IC50 = 16.5 nM T97747 C0JWL6 3008932 IC50 = 2.8 nM T97747 C0N8VX 3008933 IC50 = 41 nM T97747 CK7N8Y 3008934 IC50 = 11.1 nM T97747 CA58WE 3008935 IC50 = 15.5 nM T97747 C36JPC 3008936 IC50 = 9 nM T97747 CGU6O8 3008937 IC50 = 62 nM T97747 CUF0Z9 3009352 Ki = 5.2 nM T97747 CMK58I 3009353 Ki = 1.1 nM T97747 CPN54Q 3009354 Ki = 1.4 nM T97747 C6ZYX5 3009356 Ki = 1.6 nM T97747 CM80UB 3010250 IC50 = 6000 nM T97747 C2PNE4 3010251 IC50 = 6000 nM T97747 CB9C6Y 3010252 IC50 = 15000 nM T97747 CJBC38 3010256 IC50 = 18.1 nM T97747 C7GV5W 3010257 IC50 = 27 nM T97747 CVC2U8 3010258 IC50 = 23 nM T97747 C5XB2T 3010259 IC50 = 6.2 nM T97747 CX9PH2 3010260 IC50 = 1.1 nM T97747 CLR3U2 3010261 IC50 = 0.67 nM T97747 CIS59J 3010262 IC50 = 1.3 nM T97747 CVL16O 3010263 IC50 = 2 nM T97747 CX3IP6 3010264 IC50 = 0.2897 nM T97747 C5WT4G 3010265 IC50 = 1.5 nM T97747 CLSN01 3010266 IC50 = 7 nM T97747 C0DJQ4 3010267 IC50 = 0.73 nM T97747 C1T3CG 3010268 IC50 = 0.38 nM T97747 C7JI2E 3010269 IC50 = 3.802 nM T97747 CKS98E 3010270 IC50 = 1.6 nM T97747 CD16BY 3010271 IC50 = 0.34 nM T97747 C2TG9W 3010272 IC50 = 0.51 nM T97747 CGZV74 3010273 IC50 = 0.23 nM T97747 CC8YU9 3010274 IC50 = 0.23 nM T97747 CA2LX4 3010275 IC50 = 0.57 nM T97747 C7ON3J 3010276 IC50 = 0.6 nM T97747 CJQ5B0 3010277 IC50 = 0.89 nM T97747 CQC1H6 3010278 IC50 = 0.76 nM T97747 C4RFK6 3010279 IC50 = 0.7 nM T97747 CW3OZ1 3010280 IC50 = 1 nM T97747 C0WZ9R 3011719 IC50 = 363 nM T97747 C7SG4P 3011721 IC50 = 83 nM T97747 CFOY69 3011722 IC50 = 339 nM T97747 C5R1AW 3011723 IC50 = 8.9 nM T97747 CF53ZB 3011725 IC50 = 126 nM T97747 CSED31 3011729 IC50 = 5 nM T97747 CWOH42 3011734 IC50 = 2.4 nM T97747 C53JFX 3013575 IC50 = 5.3 nM T97747 CD5LN4 3013673 IC50 = 16 nM T97747 CZSP97 3013684 IC50 = 1.2 nM T97747 C7M4ZG 3013689 IC50 = 2.1 nM T97747 C6AV0J 3013701 IC50 = 0.8 nM T97747 CZ9M6G 3209888 IC50 = 79400 nM T97747 CNK42U 3258407 EC50 = 1900 nM T97747 CZ2G4M 4080740 IC50 = 49000 nM T97747 CKEC40 5275759 IC50 = 1.4 nM T97747 CD3C4L 5275760 IC50 = 4.6 nM T97747 C56OAD 5275761 IC50 = 44 nM T97747 C6N2GA 5275762 IC50 = 8.9 nM T97747 CE52UZ 5275763 IC50 = 5.1 nM T97747 CD9UY7 5275764 IC50 = 8.2 nM T97747 CPH85Y 5275765 IC50 = 2.2 nM T97747 C8RK0Q 5275829 IC50 = 2 nM T97747 CPUL05 5275832 IC50 = 36.7 nM T97747 CSMT51 5275833 IC50 = 350 nM T97747 CMVX10 5275835 IC50 = 11 nM T97747 CCI94R 5275836 IC50 > 2000 nM T97747 CWJC59 5275837 IC50 = 9 nM T97747 C0QK9G 5275839 IC50 = 6.4 nM T97747 CU0IJ1 5275840 IC50 = 28 nM T97747 C7UZ4T 5275841 IC50 = 10 nM T97747 CAT0F3 5275842 IC50 = 5.3 nM T97747 COFC54 5347695 IC50 > 30000 nM T97747 C04WJE 5479787 IC50 = 40 nM T97747 C9LO0F 5479840 Ki = 19 nM T97747 C59FSP 5479841 Ki = 1.1 nM T97747 CGH7F6 5479842 Ki = 3.4 nM T97747 CHXB92 5479843 Ki = 2 nM T97747 CCW7L9 5479844 Ki = 1.8 nM T97747 CQ63MB 5479845 Ki = 2 nM T97747 CS64KP 5479851 Ki = 18 nM T97747 C54DRO 5479852 Ki = 4.5 nM T97747 CMT8K7 5481702 IC50 = 10 nM T97747 C95HGD 5481703 IC50 = 15 nM T97747 CQ1WY9 5481704 IC50 = 100 nM T97747 C6DS7P 5481705 IC50 = 399.94 nM T97747 CF6W1C 5481707 IC50 = 1199.5 nM T97747 CZO76A 5481711 IC50 = 180 nM T97747 CXAK62 5481712 IC50 = 50 nM T97747 CMK83F 5481713 IC50 = 5 nM T97747 C31PZY 5481714 IC50 = 100 nM T97747 CYK98N 5481715 IC50 = 299.92 nM T97747 C7JH1S 5481716 IC50 = 100 nM T97747 CQFS90 5481726 IC50 = 120 nM T97747 C2X7VQ 5481727 IC50 = 699.84 nM T97747 CN95LU 5481736 IC50 = 640 nM T97747 CDGR53 5481737 IC50 = 780 nM T97747 C0L1UR 5481741 IC50 = 1000 nM T97747 CE3MS6 5481742 IC50 = 4 nM T97747 CUCQ49 5481743 IC50 = 4 nM T97747 C9R1OG 5481744 IC50 = 50 nM T97747 C2UG0D 5481745 IC50 = 449.78 nM T97747 C4NP6M 5481746 IC50 = 40 nM T97747 CD8H1T 5481747 IC50 = 2600.16 nM T97747 CTHN69 5481748 IC50 = 60 nM T97747 COU51D 5481749 IC50 = 5902.01 nM T97747 C01YKP 5481750 IC50 = 100 nM T97747 C1BZ4F 5481751 IC50 = 90 nM T97747 C3M6UP 5481752 IC50 = 120 nM T97747 CQTH08 5481754 IC50 = 100 nM T97747 CF5AX1 5481859 IC50 = 270 nM T97747 CD3I2R 5481861 IC50 = 270 nM T97747 C6UZJ0 5481866 IC50 = 200 nM T97747 C3HG0F 5481867 IC50 = 80 nM T97747 CZU13P 5481871 IC50 = 570 nM T97747 C3PTO2 5482298 Ki = 1.1 nM T97747 CF6PQ5 5482299 Ki = 2.2 nM T97747 CAY72C 5482300 Ki = 0.4 nM T97747 CU9D7T 5482301 Ki = 0.3 nM T97747 CSM61O 5482453 IC50 = 35 nM T97747 C6P2SJ 5482454 IC50 = 35 nM T97747 CM4SG8 5482456 IC50 = 2400 nM T97747 CR37LY 5482457 IC50 = 599.79 nM T97747 C5E4PX 5482807 IC50 = 1600 nM T97747 CSDH37 5482808 IC50 = 230 nM T97747 CMG39Z 5482809 IC50 = 10000 nM T97747 C2WV1F 5482810 IC50 = 130 nM T97747 CAY0F1 5482811 IC50 = 160 nM T97747 CLH72E 5495579 Ki = 23 nM T97747 C06TBN 5495580 Ki = 8.8 nM T97747 CZL2A6 5495581 Ki = 1.2 nM T97747 C1CBX6 5495582 Ki = 0.7 nM T97747 CZ34KJ 5495583 Ki = 4.7 nM T97747 CZMA67 5495584 Ki = 2 nM T97747 C73MGH 5495585 Ki = 14 nM T97747 CC32FY 5495586 Ki = 8.1 nM T97747 CB5ZE4 5495587 Ki = 11 nM T97747 C94XKN 5495588 Ki = 3.3 nM T97747 C94XMP 5495589 Ki = 2.1 nM T97747 CSQ6J1 5495590 Ki = 3.2 nM T97747 C3QE4X 5495591 Ki = 5.7 nM T97747 C1FJ2B 5495592 Ki = 60 nM T97747 CCD24B 5495593 Ki = 315 nM T97747 CJ02MD 5495594 Ki = 43 nM T97747 CJ6WT9 5495595 Ki = 25 nM T97747 C72OIB 5495596 Ki = 5.3 nM T97747 C6AIC7 5495597 Ki = 1.3 nM T97747 C8Q2HF 5496098 Ki = 78 nM T97747 CU45LD 5496099 Ki = 3 nM T97747 CCS5G7 5496100 Ki = 9 nM T97747 C6YTS3 5496101 Ki = 4 nM T97747 CGZ4H2 5496102 Ki = 33 nM T97747 C6U1JH 5496103 Ki = 33 nM T97747 CWK9Z7 5496104 Ki > 30 nM T97747 C9EKW0 5496105 Ki = 26 nM T97747 C3K4OF 5496106 Ki > 30 nM T97747 CJ6PF5 5496107 Ki = 7 nM T97747 CD39HS 5496108 Ki = 43 nM T97747 CNV6Y1 5496109 Ki > 30 nM T97747 C2JN1C 5496110 Ki > 30 nM T97747 C6RW0S 5496111 Ki > 30 nM T97747 CPBD91 5496112 Ki = 16 nM T97747 CCDG57 5496113 Ki = 5.3 nM T97747 C65BAI 5496114 Ki = 7.6 nM T97747 C7EQ2H 5496115 Ki = 30 nM T97747 CL9T5D 5496116 Ki = 24 nM T97747 C7QFB3 5496117 Ki = 3.8 nM T97747 C86DKQ 5496118 Ki = 4.4 nM T97747 C1VGC8 5496119 Ki = 20 nM T97747 CETR80 5496120 Ki = 5.6 nM T97747 CWLT23 5496121 Ki = 30 nM T97747 CA74LD 6320546 IC50 = 51 nM T97747 CU64LG 6320579 IC50 = 31.9 nM T97747 CHC9Y0 6320580 IC50 > 100 nM T97747 C2U7CA 6320581 IC50 = 16 nM T97747 CB41ZV 6320582 IC50 = 2 nM T97747 CLY09O 6320585 IC50 = 2 nM T97747 CY3S4K 6480206 IC50 = 32000 nM T97747 C9AFC3 6532433 Ki = 2.2 nM T97747 CD03OA 6532434 Ki = 0.4 nM T97747 CK5F9T 6532435 Ki = 0.3 nM T97747 C7J6DP 6532436 Ki = 0.1 nM T97747 C0IGN3 6533779 Ki = 2.3 nM T97747 C3E9JO 6533780 Ki = 8.8 nM T97747 CJ0I8N 6533781 Ki = 1.2 nM T97747 CHCY06 6918496 IC50 > 1000 nM T97747 C3M8YI 9574356 Ki = 18 nM T97747 CG4WA2 9574357 Ki = 1.1 nM T97747 CJN17G 9574358 Ki = 3.4 nM T97747 C59BRT 9574359 Ki = 18 nM T97747 CD2SY1 9574360 Ki = 4.5 nM T97747 C6C0XH 9575320 Ki = 1.1 nM T97747 C7GYD5 9579116 Ki = 0.7 nM T97747 C68CDO 9579117 Ki = 4.7 nM T97747 C2MV5K 9808628 IC50 = 25 nM T97747 C5T8RE 9809508 IC50 = 4.5 nM T97747 CC5EI0 9810893 IC50 = 0.24 nM T97747 CO1JI7 9827221 IC50 = 6 nM T97747 CY39ML 9869601 IC50 = 199.99 nM T97747 C9FO1Q 9873546 IC50 = 72 nM T97747 COHL06 9894474 IC50 = 240 nM T97747 C46YOP 9909684 IC50 = 6100 nM T97747 CZ7P4T 9914742 IC50 = 1.8 nM T97747 CU5O1J 9915724 IC50 = 19 nM T97747 C03TPL 9916998 IC50 = 0.22 nM T97747 CX9V2G 9917628 IC50 = 1.8 nM T97747 CSH40U 9936494 IC50 = 20 nM T97747 CQ76HK 9938497 IC50 = 43 nM T97747 C91RTG 9956238 IC50 = 400 nM T97747 C0FHY1 9978318 IC50 = 5500 nM T97747 CRP06Q 10008425 IC50 = 7.244 nM T97747 CPXO85 10008490 IC50 = 4786.3 nM T97747 C3VB2C 10008665 IC50 = 2.5 nM T97747 CVG30F 10008921 IC50 = 9120.11 nM T97747 CG1KV2 10030170 IC50 = 3 nM T97747 C1X9CD 10053691 IC50 = 1479.11 nM T97747 C4S1FH 10076141 IC50 = 0.05998 nM T97747 CRT92N 10116073 IC50 = 3000 nM T97747 C49DEF 10117347 IC50 = 120 nM T97747 C2B4CH 10118535 IC50 = 330 nM T97747 C52GKX 10143882 IC50 = 300 nM T97747 C2U4WP 10159217 IC50 = 560 nM T97747 CR2WS1 10163007 IC50 = 0.5 nM T97747 C1BGH8 10182763 IC50 = 7600 nM T97747 C2ED3X 10184169 IC50 = 2000 nM T97747 C4UC7K 10186729 IC50 = 24 nM T97747 C3DM7B 10186910 IC50 = 1.7 nM T97747 C16FPR 10187991 IC50 = 160 nM T97747 CXK43P 10204589 IC50 = 3200 nM T97747 C4OM2Z 10205915 IC50 = 3000 nM T97747 CWC7X1 10208080 IC50 = 11 nM T97747 CS27UD 10208679 IC50 = 68 nM T97747 CO2T6R 10228759 IC50 = 50 nM T97747 C72HMR 10228761 IC50 = 17 nM T97747 CE95ZB 10230510 IC50 = 229000 nM T97747 CK49NQ 10272003 IC50 = 2900 nM T97747 C3CZ7H 10277466 IC50 = 20 nM T97747 CM6SE7 10280445 IC50 = 1 nM T97747 CE9ID0 10280944 IC50 = 6.1 nM T97747 C80DZB 10290194 IC50 = 89 nM T97747 CO0P4F 10301330 IC50 = 94 nM T97747 CWFB30 10323427 IC50 > 1000 nM T97747 CFAU91 10325578 IC50 = 7 nM T97747 CRZD69 10347790 IC50 = 0.2999 nM T97747 CQP8C4 10348408 IC50 = 5 nM T97747 CPU68L 10369469 IC50 = 0.3 nM T97747 CU5F2P 10371054 IC50 = 3981.07 nM T97747 C2Y8DC 10393635 IC50 = 1023.29 nM T97747 CV60SK 10413034 IC50 = 0.9 nM T97747 CYXB38 10414981 IC50 = 0.2 nM T97747 CJ6X4K 10416552 IC50 = 20417.38 nM T97747 CZK8R4 10425374 IC50 = 154000 nM T97747 CME0U1 10438399 IC50 = 3 nM T97747 CL75IC 10445499 IC50 = 20000 nM T97747 CFD3H2 10461319 IC50 = 7 nM T97747 CI3X4T 10462202 IC50 = 1.5 nM T97747 C2D5KO 10483364 IC50 = 141.25 nM T97747 CS8A6G 10531271 IC50 = 1100 nM T97747 C2YBW0 10555236 IC50 = 660 nM T97747 C96PZF 10617034 Ki = 2 nM T97747 C2N8IQ 10627515 IC50 = 110 nM T97747 C45TVD 10648217 IC50 = 840 nM T97747 C62DKM 10650855 IC50 = 380 nM T97747 CNV4E6 10695549 IC50 = 3200 nM T97747 CT9Y3K 10698789 IC50 = 6.8 nM T97747 C1TZO6 10746493 IC50 = 1.4 nM T97747 CDLS35 10746690 IC50 = 3.1 nM T97747 CRY4I7 10747204 IC50 = 2.2 nM T97747 CCG8V9 10792796 IC50 = 570 nM T97747 C87XAH 10793079 IC50 = 1200 nM T97747 CSWN32 10840407 IC50 = 430 nM T97747 C8W7IY 10840676 IC50 = 620 nM T97747 C5XMK1 10840679 IC50 = 390 nM T97747 CJK35A 10841420 IC50 = 3.3 nM T97747 CCDO97 10842229 IC50 = 3.8 nM T97747 CW9A7C 11069824 Ki = 275 nM T97747 C15AOC 11154101 IC50 = 4700 nM T97747 CVB54S 11157818 IC50 = 60 nM T97747 C2MFC7 11166533 IC50 = 449.78 nM T97747 C7V6JL 11177360 IC50 = 149.97 nM T97747 C6FK0H 11180743 IC50 = 30 nM T97747 CI05VQ 11189082 IC50 = 49 nM T97747 C8M4RU 11192476 IC50 = 34 nM T97747 CXF20N 11193076 IC50 = 130 nM T97747 CPRH05 11204141 IC50 = 60 nM T97747 CD98SL 11204472 IC50 = 1050 nM T97747 CKO02A 11210440 IC50 = 599.79 nM T97747 C2RBU8 11215601 IC50 = 50 nM T97747 CIS29O 11215950 IC50 = 89 nM T97747 CZ20TE 11224188 IC50 = 10100 nM T97747 CA39QR 11227406 IC50 > 1000 nM T97747 CN84TM 11234566 IC50 = 40000 nM T97747 CN51JH 11238728 IC50 = 50 nM T97747 C21OTD 11246827 IC50 = 149.97 nM T97747 CAR46F 11249997 IC50 = 4800 nM T97747 CS9I8P 11250534 IC50 = 70 nM T97747 CA5ST9 11259200 IC50 = 8500 nM T97747 C31MVR 11261876 IC50 = 40 nM T97747 CQ6KW0 11272103 IC50 = 1000 nM T97747 C06TUD 11285791 IC50 = 0.1 nM T97747 C5DG8M 11326950 IC50 = 349.95 nM T97747 C1A5ET 11329244 IC50 = 1000 nM T97747 CI3YG0 11342750 IC50 = 68 nM T97747 C5LK1F 11342841 IC50 = 25 nM T97747 C74ZPM 11350639 IC50 = 1400 nM T97747 CSAD06 11353001 IC50 = 1.1 nM T97747 CCZN17 11365412 IC50 = 40 nM T97747 CBZ18L 11376667 IC50 = 50 nM T97747 C8DJL6 11399408 IC50 = 30 nM T97747 C6RQ0D 11408704 IC50 = 1300 nM T97747 C5UZ6O 11410758 IC50 = 130 nM T97747 C7T9JS 11421221 IC50 = 13 nM T97747 C19RCV 11422270 IC50 = 30 nM T97747 C1E6KF 11433338 IC50 = 26 nM T97747 C6VCP5 11433740 IC50 = 30 nM T97747 CBEF39 11444710 IC50 = 140 nM T97747 CS6LA7 11466794 IC50 = 19 nM T97747 C7Z9KU 11467704 IC50 = 1.995 nM T97747 C6ZI2E 11478988 IC50 = 40 nM T97747 CW6YN0 11490468 IC50 = 140 nM T97747 C40IMW 11502371 IC50 = 1000 nM T97747 CA3SW7 11503459 IC50 = 2 nM T97747 CGN4S8 11505350 IC50 = 1.7 nM T97747 C3LBY6 11513274 IC50 = 0.21 nM T97747 C8P4GL 11520480 IC50 = 25 nM T97747 C4XVL8 11520510 IC50 = 67 nM T97747 CYH8J9 11525100 IC50 = 1.2 nM T97747 C7HF1B 11527582 IC50 = 12 nM T97747 C7LP9F 11527691 IC50 = 4.7 nM T97747 C0F7SR 11534473 IC50 = 1610 nM T97747 C0NL5U 11569805 IC50 = 84 nM T97747 CLY5O2 11570431 IC50 = 220 nM T97747 CE5KD2 11570778 IC50 = 2.8 nM T97747 C70EYD 11577846 IC50 = 3.2 nM T97747 C4KQI5 11578088 IC50 = 730 nM T97747 CAS56U 11585418 IC50 = 3.9 nM T97747 CEC49G 11585625 IC50 = 4.1 nM T97747 C1DKF4 11598797 IC50 = 610 nM T97747 CJ1IF0 11605997 IC50 = 1.2 nM T97747 C84YPR 11606411 IC50 = 630 nM T97747 C7C8FX 11626984 IC50 = 9 nM T97747 C57RHQ 11634966 IC50 = 860 nM T97747 C9CKA0 11635721 IC50 = 1.7 nM T97747 C54OFG 11636141 IC50 = 0.95 nM T97747 CJ3I2L 11639993 IC50 > 1000 nM T97747 CZ1T4W 11641131 IC50 = 8 nM T97747 C0XZK5 11650548 IC50 = 0.19 nM T97747 CH97IX 11656080 IC50 = 21.5 nM T97747 CU7OG2 11669935 IC50 = 283 nM T97747 CFV0I9 11690481 IC50 = 17 nM T97747 CPIY98 11692945 IC50 = 6.4 nM T97747 C6WD8L 11693007 IC50 = 20 nM T97747 C17RPK 11700429 IC50 = 0.48 nM T97747 CCG50D 11753754 IC50 = 190 nM T97747 CHS9Q3 11785237 IC50 < 0.1 nM T97747 CFA15U 11786927 IC50 = 10 nM T97747 C9OTN2 11787124 IC50 = 76 nM T97747 C2J8RH 11844212 IC50 = 30 nM T97747 CL1FX0 11947758 IC50 = 380.19 nM T97747 CGP04N 11988311 IC50 = 0.137 nM T97747 CJX31Q 12093170 IC50 = 703 nM T97747 CK80NA 12987698 EC50 = 1900 nM T97747 CJGC50 14434082 EC50 = 10000 nM T97747 C8L9VX 15485365 IC50 = 1000 nM T97747 CIZ8C1 15783796 EC50 = 1995.26 nM T97747 CCDX50 15940498 IC50 = 0.5 nM T97747 CU02IX 15940799 IC50 = 0.3 nM T97747 CN4F8X 15940800 IC50 = 0.1 nM T97747 C8JIP7 15940801 IC50 = 0.4 nM T97747 CTH2A9 15941083 IC50 = 0.4 nM T97747 CF30UM 15941086 IC50 = 0.1 nM T97747 CM10PF 15941255 IC50 = 0.08 nM T97747 C5WUJ0 15942352 IC50 = 48.4 nM T97747 CB8H6M 15947119 IC50 = 0.2 nM T97747 C3UW0T 15950679 IC50 = 18.9 nM T97747 C2U1GH 15958353 IC50 = 20 nM T97747 CCL59Z 16007088 IC50 = 0.32 nM T97747 CXBD17 16041224 IC50 = 6.6 nM T97747 CDU1L0 16041411 IC50 = 0.9 nM T97747 CGM4N8 16041594 IC50 = 15.7 nM T97747 CYA3K5 16064151 IC50 = 10 nM T97747 C38DNF 16073659 IC50 = 780 nM T97747 CZ5JG1 16073660 IC50 = 0.76 nM T97747 CQI01L 16073661 IC50 = 46 nM T97747 CS48RO 16073662 IC50 = 1 nM T97747 C71ODK 16073663 IC50 = 21 nM T97747 C05TIF 16073664 IC50 = 132 nM T97747 C36HRZ 16073665 IC50 = 20 nM T97747 C74ROH 16073666 IC50 = 25 nM T97747 CAK3O1 16073667 IC50 = 20 nM T97747 CO0J6E 16073668 IC50 = 560 nM T97747 C63SFG 16073669 IC50 = 32 nM T97747 CLM4I9 16073670 IC50 = 1.1 nM T97747 C3W6XJ 16073671 IC50 = 500 nM T97747 C3P8HL 16073672 IC50 = 110 nM T97747 CIWA92 16073673 IC50 = 56 nM T97747 C3Y0MT 16073674 IC50 = 25 nM T97747 C9G8TZ 16124598 IC50 = 251.19 nM T97747 CI32YP 16301115 EC50 = 13500 nM T97747 CUTB83 16655051 IC50 = 92.9 nM T97747 C3WX9K 16658855 IC50 = 6530 nM T97747 C7X0TS 16659334 IC50 = 3.5 nM T97747 CG7MA3 16726107 EC50 = 1100 nM T97747 CM0QJ2 16728324 IC50 = 8.75 nM T97747 CIFJ10 16728325 IC50 = 6.22 nM T97747 C3TNU9 16728326 IC50 = 122 nM T97747 C8UMZ1 16728609 IC50 = 599.79 nM T97747 C2YBX3 16728610 IC50 = 1900 nM T97747 C49PQF 16728611 IC50 = 800 nM T97747 CV9ZH3 16728612 IC50 = 600 nM T97747 CZ9TG7 16728613 IC50 = 480 nM T97747 C9CKU7 16728614 IC50 = 1999.86 nM T97747 CZV0H1 16728615 IC50 = 899.5 nM T97747 CGSC15 16728616 IC50 = 1698.24 nM T97747 CV54TY 16728617 IC50 = 5700 nM T97747 CJ1YK4 16728618 IC50 = 1300 nM T97747 CIM1Z9 16728619 IC50 = 1599.56 nM T97747 CY97UR 16728620 IC50 = 39000 nM T97747 C8H9RN 16728621 IC50 = 500.03 nM T97747 CUC7B5 16728622 IC50 = 1698.24 nM T97747 CED81G 16728623 IC50 = 699.84 nM T97747 CB45LR 16728624 IC50 = 2897.34 nM T97747 C9BHE4 16728625 IC50 = 1698.24 nM T97747 C8X7LT 16728626 IC50 = 1100 nM T97747 C6KDW9 16728627 IC50 = 3700 nM T97747 C3UN0X 16728628 IC50 = 8700 nM T97747 CHBQ91 16728629 IC50 = 600 nM T97747 C58IKH 16728630 IC50 = 1199.5 nM T97747 CE51NB 16728631 IC50 = 3404.08 nM T97747 C7JDU0 16728632 IC50 = 3100 nM T97747 CMG1V0 16728633 IC50 > 30000 nM T97747 C1W2VH 16728634 IC50 > 30000 nM T97747 CHQO72 16728635 IC50 = 600 nM T97747 CT7G2R 16728636 IC50 > 30000 nM T97747 CW10DK 16728637 IC50 > 30000 nM T97747 CUP1Q0 16728638 IC50 > 30000 nM T97747 C4EG0L 16728639 IC50 > 30000 nM T97747 CQP2C6 16728640 IC50 > 30000 nM T97747 CWK46L 16728641 IC50 > 30000 nM T97747 C2V1FK 16728642 IC50 = 8500 nM T97747 CD8U4Z 16728643 IC50 = 139.96 nM T97747 CS9FH8 16728644 IC50 = 399.94 nM T97747 C6LWX7 16728645 IC50 = 4197.59 nM T97747 CZU94T 16728646 IC50 > 30000 nM T97747 CD6AM7 16728647 IC50 = 749.89 nM T97747 C0CU2F 16728648 IC50 = 14000 nM T97747 CL9N1W 16728649 IC50 = 1999.86 nM T97747 C0E3SL 16728783 IC50 > 3000 nM T97747 CS1F3B 16728784 IC50 = 28 nM T97747 CFCV60 16728785 IC50 = 130 nM T97747 CDMA29 16728786 IC50 = 53 nM T97747 CAX2B7 16728787 IC50 = 1.1 nM T97747 CQ7G2U 16728788 EC50 = 2000 nM T97747 C9H8IS 16730521 IC50 = 11 nM T97747 CP4CY0 18442936 IC50 = 37 nM T97747 CTM71O 20664115 IC50 = 12 nM T97747 CES60Q 20664141 IC50 = 7 nM T97747 CB36XZ 20664149 IC50 = 0.8 nM T97747 CXOS35 20664156 IC50 = 2.5 nM T97747 C7RO9I 20664159 IC50 = 8.2 nM T97747 C87RFX 20664160 IC50 = 65 nM T97747 CFQM24 20664161 IC50 = 0.42 nM T97747 CUZ8P0 20664163 IC50 = 2.799 nM T97747 CBJ5N8 20672360 IC50 = 0.5 nM T97747 CLE46M 20672362 IC50 = 0.3 nM T97747 CS20IY 20672370 IC50 = 0.3 nM T97747 CJXP29 20672384 IC50 = 0.84 nM T97747 C2DEH4 20672386 IC50 = 0.5 nM T97747 C2PG9O 21064126 IC50 = 79 nM T97747 CFWJ06 21064281 IC50 = 28 nM T97747 CHC4Q3 21064283 IC50 = 13 nM T97747 CS78PF 21064289 IC50 = 92 nM T97747 C3K0IQ 21064293 IC50 = 130 nM T97747 CDU03R 21064295 IC50 = 33 nM T97747 C5R4DC 21064297 IC50 = 79 nM T97747 CND40Q 21064299 IC50 = 40 nM T97747 CS6IT0 21064329 IC50 = 86 nM T97747 CTMC32 21064331 IC50 = 170 nM T97747 CA1E0H 21064338 IC50 = 450 nM T97747 C8NTA6 21147749 IC50 = 2 nM T97747 CY0J1U 21148035 IC50 = 1000 nM T97747 CE38ZB 21341080 IC50 = 1.6 nM T97747 C9YZ3A 21867666 IC50 = 7 nM T97747 CKGT37 21925890 IC50 = 570 nM T97747 CE05FA 21926122 IC50 > 3000 nM T97747 C4WX7Q 21926246 IC50 > 3000 nM T97747 C0UT7V 21926618 IC50 = 69 nM T97747 CWH1D9 21926948 IC50 = 52 nM T97747 C3E0DK 21927225 IC50 = 54 nM T97747 CE2P5B 21927257 IC50 = 590 nM T97747 CO9VD3 22135856 IC50 > 3000 nM T97747 C8HE4I 23285265 IC50 = 720 nM T97747 CXF8Z9 23294208 IC50 = 19952.62 nM T97747 C3XN1D 23294214 IC50 = 1584.89 nM T97747 C32CYE 23577328 IC50 = 33000 nM T97747 CQ4M2S 23577360 IC50 = 39000 nM T97747 C1VX7E 23577362 IC50 = 3500 nM T97747 C6P2HL 23577370 IC50 = 2800 nM T97747 C5ZSO4 23577378 IC50 = 7100 nM T97747 CAX0O6 23577382 IC50 = 7400 nM T97747 C3U9PK 23577386 IC50 = 1400 nM T97747 C7SD8Q 23577388 IC50 = 34000 nM T97747 C16ZJO 23577409 IC50 = 13000 nM T97747 C6SB3P 23577448 IC50 = 30000 nM T97747 CP2RA0 23577500 IC50 > 3000 nM T97747 CE29IW 23650547 IC50 = 1 nM T97747 C7JV4W 23725177 IC50 = 780 nM T97747 C25HKJ 24758044 IC50 > 20000 nM T97747 C4AEG2 25024699 IC50 = 1.7 nM T97747 C5M2CK 25057602 IC50 = 144 nM T97747 C91NVS 25057877 IC50 = 300 nM T97747 C6MO8Z 25130569 IC50 = 3467.37 nM T97747 CUH0C9 25130571 IC50 = 9332.54 nM T97747 C4MR8V 25130901 IC50 = 776.25 nM T97747 CE30DM 25130903 IC50 = 5248.07 nM T97747 CO4VZ3 25130904 IC50 > 31622.78 nM T97747 C4OY2V 25131220 IC50 > 31622.78 nM T97747 C0J1OY 25131899 IC50 > 31622.78 nM T97747 C3N2LV 25131900 IC50 = 19952.62 nM T97747 CCPA34 25131901 IC50 = 1258.93 nM T97747 CJG1U8 25131902 IC50 = 3981.07 nM T97747 CWA93M 25132253 IC50 = 63.1 nM T97747 C3I1XJ 25132254 IC50 = 5.012 nM T97747 CY52ZQ 25132255 IC50 = 19.95 nM T97747 CM30EC 25132603 IC50 = 1 nM T97747 CK0L3W 25132604 IC50 = 5.012 nM T97747 C4GF3T 25132945 IC50 = 2398.83 nM T97747 C1WAP7 25132946 IC50 = 9332.54 nM T97747 CY8R6L 25132948 IC50 > 31622.78 nM T97747 COK24W 25133270 IC50 = 7079.46 nM T97747 CGR54C 25133271 IC50 = 446.68 nM T97747 CTQ2C7 25133617 IC50 = 5011.87 nM T97747 C8R5JI 25133618 IC50 = 7943.28 nM T97747 C28FCZ 25133619 IC50 = 8511.38 nM T97747 C9PCN5 25133620 IC50 = 4570.88 nM T97747 CQ4ZJ9 25133961 IC50 = 63.1 nM T97747 C0XNZ7 25133962 IC50 = 15.85 nM T97747 CIY4Q3 25133963 IC50 = 5.248 nM T97747 C2LZN5 25133964 IC50 = 29.51 nM T97747 C54KPB 25205600 IC50 = 65 nM T97747 C6J3TG 25205601 IC50 = 84 nM T97747 CE0WO1 25205764 IC50 = 43 nM T97747 CR49UP 25205766 IC50 = 20 nM T97747 CV02HS 25205767 IC50 = 12 nM T97747 CBH92X 25205921 IC50 = 27 nM T97747 C84EQC 25205923 IC50 = 6 nM T97747 CH4ZW0 25206069 IC50 = 90 nM T97747 CW0FH8 25206070 IC50 = 21 nM T97747 C6HWA7 25206071 IC50 = 26 nM T97747 C2K9DX 25206204 IC50 = 60 nM T97747 C13FTZ 25206227 IC50 = 34 nM T97747 C0VWM1 25206397 IC50 = 32 nM T97747 C2GU6Q 25230769 IC50 > 500 nM T97747 C7SUF3 25230770 IC50 = 217 nM T97747 CQP83X 25230771 IC50 = 19 nM T97747 CRCS05 25230773 IC50 = 19 nM T97747 CO9T8A 25230826 IC50 = 18 nM T97747 C8WF3A 25230827 IC50 = 22 nM T97747 C54LQF 25230828 IC50 = 30 nM T97747 CR31QN 25230829 IC50 = 25 nM T97747 C2M8SR 25230896 IC50 = 349 nM T97747 CT21IO 25230897 IC50 = 60 nM T97747 CB9V4X 25230898 IC50 = 22 nM T97747 CH6N1A 25230899 IC50 = 27 nM T97747 CKH70V 25230969 IC50 > 500 nM T97747 CVXD97 25230970 IC50 = 11 nM T97747 CU1W0E 25230971 IC50 = 80 nM T97747 CJ54KN 25231038 IC50 = 70 nM T97747 CV2L4K 25231041 IC50 = 64 nM T97747 COQI09 25231105 IC50 = 78 nM T97747 CBMH73 25256856 IC50 = 2 nM T97747 CJ0ZN4 25256857 IC50 = 8 nM T97747 C2FZ9P 42606792 IC50 = 1636 nM T97747 CI1C5U 42623163 IC50 = 2 nM T97747 C4HL1I 44129650 IC50 = 37.3 nM T97747 CEKX13 44194496 IC50 = 113.6 nM T97747 CV9M8D 44194587 IC50 = 3.32 nM T97747 C4AZ9G 44194588 IC50 = 1.53 nM T97747 C0Q5SE 44194589 IC50 = 2.1 nM T97747 CY0V2U 44194590 IC50 = 1.09 nM T97747 CM7OY9 44194675 IC50 = 5 nM T97747 C4BJA6 44194676 IC50 = 2.93 nM T97747 C1PT3U 44205000 IC50 = 0.9 nM T97747 C5YFB9 44252324 IC50 > 10000 nM T97747 CM67JX 44273531 IC50 = 0.1 nM T97747 CEF2O4 44273816 IC50 = 1.1 nM T97747 C7P5EI 44273830 IC50 = 0.2 nM T97747 COX48Y 44273846 IC50 = 1000 nM T97747 CJ4H3K 44273850 IC50 = 51 nM T97747 CY31BC 44273872 IC50 = 1.5 nM T97747 C1G9IF 44273888 IC50 = 0.4 nM T97747 CG46IJ 44273960 IC50 = 0.7998 nM T97747 CU5O9Q 44273996 IC50 = 0.4 nM T97747 CO8VE2 44274022 IC50 = 3.7 nM T97747 C7MZA3 44274042 IC50 = 4.797 nM T97747 CTB92I 44274043 IC50 = 0.2 nM T97747 CJOD81 44274090 IC50 = 1.6 nM T97747 CG8A6Y 44274106 IC50 = 0.9 nM T97747 CM4VI3 44274108 IC50 = 0.8 nM T97747 CW5KM0 44322729 IC50 = 70 nM T97747 CN3YT4 44324386 IC50 = 4000 nM T97747 CV1G7P 44325489 IC50 = 19 nM T97747 CY3L7S 44325511 IC50 = 220 nM T97747 CJC29B 44325542 IC50 = 4 nM T97747 C5BJ1O 44325665 IC50 = 0.8 nM T97747 CW36ZF 44325710 IC50 = 22 nM T97747 C47CDP 44325917 IC50 = 22 nM T97747 CTL92Q 44332341 IC50 = 0.2 nM T97747 C7SNJ5 44332489 IC50 = 0.4 nM T97747 C03NLX 44332684 IC50 = 0.1 nM T97747 CQT3M4 44332814 IC50 = 1 nM T97747 CJQA92 44335765 IC50 = 10 nM T97747 C2TEM7 44336415 IC50 = 20 nM T97747 CPGN89 44337326 Ki = 1 nM T97747 C5OE3P 44341106 Ki = 2 nM T97747 C0K5BM 44342961 IC50 = 0.23 nM T97747 CED6Z5 44342962 IC50 = 0.23 nM T97747 C8ON9S 44356876 IC50 = 21 nM T97747 C60YTZ 44356944 IC50 = 1.5 nM T97747 CHN56D 44356952 IC50 = 1.2 nM T97747 CBFY26 44357063 IC50 = 1.2 nM T97747 CSL5R9 44357072 IC50 = 0.8 nM T97747 CHM12S 44357078 IC50 = 0.5 nM T97747 C64KXD 44357079 IC50 = 0.4 nM T97747 CK9G2U 44357375 IC50 = 1.7 nM T97747 C7CMB3 44357379 IC50 = 1.1 nM T97747 CZTI85 44373672 IC50 = 27 nM T97747 C48ELJ 44373721 IC50 = 5 nM T97747 CDP34B 44373748 IC50 = 86 nM T97747 CZU19Q 44373755 IC50 ~ 27 nM T97747 CWM1F5 44373756 IC50 = 0.13 nM T97747 CJ6X0R 44373767 IC50 = 69 nM T97747 C5F3AQ 44373768 IC50 = 33 nM T97747 C0I1AL 44373852 IC50 = 5 nM T97747 C4QN7Z 44373926 IC50 = 6 nM T97747 CD64UI 44373973 IC50 = 14 nM T97747 C4ZCA2 44374016 IC50 = 8 nM T97747 CHD26R 44374017 IC50 = 43 nM T97747 CG14HU 44374086 IC50 = 30 nM T97747 C4B8ZF 44374088 IC50 = 11 nM T97747 COT83J 44374136 IC50 = 46 nM T97747 C76UBK 44383760 IC50 = 41 nM T97747 C60VEP 44383787 IC50 = 2.1 nM T97747 C74DCF 44384011 IC50 = 11.5 nM T97747 C09IYH 44384012 IC50 = 23 nM T97747 C4A3GF 44384584 IC50 = 1 nM T97747 CCK72Y 44384642 IC50 = 4.4 nM T97747 CE0S9Q 44384705 IC50 = 6.9 nM T97747 CG9K8P 44384782 IC50 = 0.5 nM T97747 CH6J3Q 44384875 IC50 = 1.2 nM T97747 CO9P8X 44384927 IC50 = 0.8 nM T97747 C3QL8D 44384969 IC50 = 11 nM T97747 CUCH65 44385583 IC50 = 0.5 nM T97747 CQ58FI 44389412 IC50 = 3.6 nM T97747 C4PH3E 44392074 IC50 = 91 nM T97747 C8UZX0 44392078 IC50 = 8700 nM T97747 CHMY61 44392082 IC50 = 3600 nM T97747 CDN01K 44392083 IC50 = 3500 nM T97747 CWJK96 44392084 IC50 = 690 nM T97747 C2VN8S 44392087 IC50 < 10 nM T97747 CN0H4K 44392088 IC50 = 46 nM T97747 C8B9XD 44392092 IC50 = 2200 nM T97747 CM5F6G 44392093 IC50 = 2300 nM T97747 C3E6SV 44392094 IC50 = 180 nM T97747 CWY84B 44392095 IC50 = 7900 nM T97747 C27ISR 44392096 IC50 = 76 nM T97747 C91WEC 44392103 IC50 = 630 nM T97747 CC8L5E 44392104 IC50 = 4900 nM T97747 CR5NG8 44392105 IC50 = 800 nM T97747 C98EUH 44392106 IC50 = 370 nM T97747 C98COA 44392109 IC50 = 5500 nM T97747 CZ1A4U 44392110 IC50 = 580 nM T97747 C4CHI6 44392111 IC50 = 110 nM T97747 CH90MX 44392114 IC50 = 470 nM T97747 CT3V8A 44392115 IC50 = 5900 nM T97747 CXU52S 44392116 IC50 = 780 nM T97747 C7MIY0 44392117 IC50 = 290 nM T97747 CI5S1Q 44392123 IC50 = 770 nM T97747 CQ3UK0 44392124 IC50 = 650 nM T97747 CIHT56 44392125 IC50 = 33 nM T97747 CAS85F 44392126 IC50 = 4100 nM T97747 C2G1OP 44392130 IC50 = 150 nM T97747 C4F9EW 44392131 IC50 = 2100 nM T97747 CN3B8U 44392132 IC50 = 2600 nM T97747 C9O8VP 44392135 IC50 = 5900 nM T97747 CX69VZ 44392136 IC50 = 2700 nM T97747 CXO91S 44392137 IC50 = 32 nM T97747 C6X1LF 44392142 IC50 = 310 nM T97747 CZOV60 44392143 IC50 = 370 nM T97747 CM83HG 44392144 IC50 = 1900 nM T97747 C4H0PT 44392147 IC50 = 1100 nM T97747 C3PHL1 44392148 IC50 = 680 nM T97747 CK27GP 44392149 IC50 = 310 nM T97747 C7KXJ0 44392153 IC50 = 66 nM T97747 CMZ6P9 44392154 IC50 = 7200 nM T97747 CGU0F6 44392155 IC50 = 1400 nM T97747 CCTR59 44392159 IC50 = 190 nM T97747 C3TCB0 44392160 IC50 = 6800 nM T97747 CXZU54 44392161 IC50 = 60 nM T97747 C0MN1I 44392162 IC50 = 350 nM T97747 C72VXL 44392166 IC50 = 580 nM T97747 CR4JP7 44392167 IC50 = 38 nM T97747 C31FMI 44392168 IC50 = 5100 nM T97747 CXUA20 44392169 IC50 = 660 nM T97747 CQTD48 44392176 IC50 = 49 nM T97747 CJ4QA3 44392196 IC50 = 240 nM T97747 C3QNW5 44392203 IC50 = 680 nM T97747 C70TGZ 44392204 IC50 = 560 nM T97747 C9BM2F 44392211 IC50 = 1800 nM T97747 CQWI02 44392213 IC50 = 320 nM T97747 CY5TX7 44392218 IC50 = 7400 nM T97747 CV41WR 44392219 IC50 = 3400 nM T97747 CMVR86 44392220 IC50 = 110 nM T97747 CAZ5I4 44392229 IC50 = 100 nM T97747 CSNB94 44392235 IC50 = 35 nM T97747 CHU5K6 44392244 IC50 = 62 nM T97747 CBA56P 44392253 IC50 = 42 nM T97747 CHT1S5 44392258 IC50 = 5400 nM T97747 CO5D7H 44395365 IC50 = 7200 nM T97747 CEY49R 44395386 IC50 = 8800 nM T97747 C0ZFD8 44401488 IC50 = 0.35 nM T97747 CHQY70 44401593 IC50 = 63 nM T97747 CL24ST 44401608 IC50 = 200 nM T97747 CQC16I 44401686 IC50 = 2.6 nM T97747 CFR53O 44401731 IC50 = 10 nM T97747 CEKA14 44401734 IC50 = 100 nM T97747 CATD12 44401751 IC50 = 0.89 nM T97747 C16MBG 44401760 IC50 = 0.82 nM T97747 CWH26M 44401763 IC50 = 12 nM T97747 CD3X4N 44401765 IC50 = 6.3 nM T97747 CH65CZ 44401863 IC50 = 12 nM T97747 CT9XO0 44401956 IC50 = 0.5 nM T97747 CJ9FS4 44401965 IC50 = 0.6 nM T97747 C8WV0Q 44401985 IC50 = 23 nM T97747 CQ6SO2 44404596 IC50 = 8.5 nM T97747 C15PRG 44404601 IC50 = 760 nM T97747 CA15WI 44404605 IC50 = 310 nM T97747 CL86FA 44404638 IC50 = 200 nM T97747 CTM2X0 44404639 IC50 = 26 nM T97747 C98QDP 44404640 IC50 = 5.9 nM T97747 CGD3Z5 44404641 IC50 = 130 nM T97747 CTC28Z 44404642 IC50 = 22 nM T97747 C34CQF 44404643 IC50 = 24 nM T97747 CVK07T 44404644 IC50 = 11 nM T97747 CMCP98 44404645 IC50 = 740 nM T97747 CZI0D9 44404650 IC50 = 19 nM T97747 CSY85U 44404656 IC50 = 105 nM T97747 CO28NW 44404657 IC50 = 7.9 nM T97747 C0J5YT 44404658 IC50 = 9.1 nM T97747 CE0CM4 44404692 IC50 = 58 nM T97747 CN30IB 44404697 IC50 = 78 nM T97747 CTFY36 44404702 IC50 = 28 nM T97747 C1CBI7 44404705 IC50 = 2.3 nM T97747 CM50EI 44404709 IC50 = 7.1 nM T97747 C5VJ9P 44404710 IC50 = 260 nM T97747 C6RAG1 44404716 IC50 < 1 nM T97747 CH3NG1 44404719 IC50 = 6.3 nM T97747 C01ZEW 44404720 IC50 = 85 nM T97747 CU9BI1 44404724 IC50 = 12 nM T97747 CD3X0F 44404730 IC50 = 200 nM T97747 CV9YH2 44412984 IC50 = 40 nM T97747 C4LT3K 44415740 IC50 = 20 nM T97747 C5U1EA 44415755 IC50 = 0.7 nM T97747 CUG6N2 44415756 IC50 = 250 nM T97747 CHU9Y6 44415783 IC50 = 70 nM T97747 C1NGI4 44415784 IC50 = 50 nM T97747 C9GO0B 44415800 IC50 = 2 nM T97747 C64VRB 44415820 IC50 = 6 nM T97747 CRJ70D 44415821 IC50 = 39 nM T97747 CT73JO 44415847 IC50 = 5 nM T97747 CMA02E 44431926 IC50 = 1300 nM T97747 CTO19K 44431931 IC50 > 30000 nM T97747 C4RST8 44431934 IC50 > 30000 nM T97747 CZ4YP3 44431944 IC50 = 279.9 nM T97747 CVMN01 44431946 IC50 = 3097.42 nM T97747 CHL9M6 44431949 IC50 = 389.94 nM T97747 CXY1F8 44431951 IC50 = 400 nM T97747 CK65WG 44431953 IC50 = 1300 nM T97747 C3E5DV 44431954 IC50 = 349.95 nM T97747 CV5CN0 44431959 IC50 = 579.43 nM T97747 C3UJ8R 44431962 IC50 = 579.43 nM T97747 C60EHY 44431965 IC50 = 1099.01 nM T97747 C7OVB6 44431967 IC50 = 210 nM T97747 C40LUV 44431969 IC50 = 1500 nM T97747 CG2AB4 44431971 IC50 = 320 nM T97747 C2SVT3 44431972 IC50 = 57 nM T97747 CQED73 44431975 IC50 = 450 nM T97747 C9JM4F 44431976 IC50 = 170 nM T97747 C80MVI 44431977 IC50 = 100 nM T97747 C7P2RW 44431979 IC50 = 47 nM T97747 C8XTN1 44431984 IC50 = 35 nM T97747 CHK5S9 44431986 IC50 = 27 nM T97747 CT93GC 44439155 IC50 = 63 nM T97747 CJPR21 44439313 IC50 = 93 nM T97747 CXU41O 44439314 IC50 = 400 nM T97747 CDFP30 44447731 IC50 = 2 nM T97747 CFAL15 44447732 IC50 = 1.3 nM T97747 C9EM8Q 44447733 IC50 = 6.5 nM T97747 CX89DC 44447734 IC50 = 0.8 nM T97747 CHKC89 44447735 IC50 = 1.8 nM T97747 CWB20Y 44454972 IC50 = 48 nM T97747 C4KX7W 44454975 IC50 = 539 nM T97747 CJZ7N1 44454977 IC50 = 4 nM T97747 C6RQY0 44454999 IC50 = 15 nM T97747 C06XYR 44455001 IC50 = 100 nM T97747 C2G0ZQ 44455031 IC50 = 27 nM T97747 CD12BW 44455033 IC50 = 53 nM T97747 C3FE8U 44455034 IC50 = 381 nM T97747 C4TFR9 44455069 IC50 = 4 nM T97747 CMF34Z 44455072 IC50 = 29 nM T97747 C3BVO1 44455103 IC50 = 271 nM T97747 CTU7H3 44455106 IC50 = 323 nM T97747 CY40FE 44455143 IC50 = 96 nM T97747 CW96PA 44455144 IC50 = 20 nM T97747 CNZ60R 44455177 IC50 = 271 nM T97747 C70PHB 44455180 IC50 = 78 nM T97747 CL12VU 44455217 IC50 = 0.4 nM T97747 C7KS8J 44455223 IC50 = 31 nM T97747 C7C1PI 44455225 IC50 = 310 nM T97747 CCA13O 44455313 IC50 = 970 nM T97747 CHEP83 44461014 IC50 > 10000 nM T97747 CME3S8 44461016 IC50 > 10000 nM T97747 CUX8D6 44461274 IC50 = 6 nM T97747 C7LQY9 44461275 IC50 = 3 nM T97747 CY32GT 44461476 IC50 = 5 nM T97747 C8JY5Z 44461494 IC50 = 35 nM T97747 CL5AM7 44461513 IC50 = 40 nM T97747 C31UNS 44461521 IC50 = 15 nM T97747 CE62UH 44461522 IC50 = 20 nM T97747 C3OTS5 44461559 IC50 = 15 nM T97747 COQZ58 44461560 IC50 = 100 nM T97747 CVC83W 44461561 IC50 = 25 nM T97747 CRZ8B2 44461581 IC50 = 39.81 nM T97747 CZH18E 44461603 IC50 = 35 nM T97747 C7PD1X 44461623 IC50 = 120 nM T97747 C2VW8I 44461628 IC50 = 10 nM T97747 CQ5XM0 44461677 IC50 = 5 nM T97747 CHC7O1 44461684 IC50 = 2 nM T97747 C3KMA9 44461689 IC50 = 4 nM T97747 CR8L1S 44461699 IC50 = 3 nM T97747 CXHT47 44461707 IC50 = 2 nM T97747 CD2KC6 44461713 IC50 = 6 nM T97747 CREY18 44461714 IC50 = 10 nM T97747 CT78IZ 44461741 IC50 = 0.75 nM T97747 CSR9Q6 44461774 IC50 = 150 nM T97747 C30PZS 44461785 IC50 = 1000 nM T97747 C5MR0E 44461790 IC50 = 1000 nM T97747 C49OIF 44461804 IC50 = 794.33 nM T97747 CZ7IX1 44461817 IC50 = 3 nM T97747 CO9RF0 44461823 IC50 = 4 nM T97747 C3XIJ9 44461831 IC50 = 100 nM T97747 CG65UL 44461835 IC50 = 20 nM T97747 C3KJP5 44511861 IC50 = 40 nM T97747 C4N5ET 44511871 IC50 = 0.8 nM T97747 C3M8UD 44511934 IC50 = 0.3 nM T97747 C2ZFD8 44511935 IC50 = 0.6 nM T97747 COK7H1 44511938 IC50 = 0.3 nM T97747 CY9FT7 44511966 IC50 = 7 nM T97747 CHV3I6 44511967 IC50 = 10.9 nM T97747 CBSD16 44512001 IC50 = 0.7 nM T97747 CM85OE 44512058 IC50 = 0.3 nM T97747 CI4S8C 44512090 IC50 = 0.3 nM T97747 C6WH8N 44512349 IC50 = 1.3 nM T97747 CGM39D 44532866 IC50 = 265 nM T97747 CT5N4E 44555481 IC50 = 4 nM T97747 C7WO5E 44555482 IC50 = 27 nM T97747 CT8S2U 44559501 IC50 = 60000 nM T97747 CF1C8U 44564835 IC50 = 89.2 nM T97747 CL4N5D 44564884 IC50 = 85.3 nM T97747 C6P8OF 44564885 IC50 = 52.8 nM T97747 CK49AW 44564886 IC50 = 3.16 nM T97747 C8URX2 44564887 IC50 = 3.11 nM T97747 CA96BX 44564929 IC50 = 3.93 nM T97747 CJ0C6T 44564930 IC50 = 0.513 nM T97747 C5AVF0 44564931 IC50 = 164 nM T97747 C5U0TR 44564982 IC50 = 4.87 nM T97747 C8GCQ6 44564983 IC50 = 6.12 nM T97747 CE1OG0 44564984 IC50 = 28.7 nM T97747 CM4Z0V 44564985 IC50 = 315 nM T97747 C9JI2F 44565035 IC50 = 176 nM T97747 C37WSJ 44565036 IC50 = 187 nM T97747 CMOC65 44565037 IC50 = 0.84 nM T97747 CG2UO0 44565038 IC50 = 0.38 nM T97747 C3MNR0 44565080 IC50 = 0.48 nM T97747 CF6JG1 44565081 IC50 = 49.9 nM T97747 CA0FC1 44565082 IC50 = 1.3 nM T97747 C6DI0T 44565083 IC50 = 62 nM T97747 C8XF4D 44565557 IC50 = 3.499 nM T97747 CXT21C 44565558 IC50 = 28.97 nM T97747 C8BL9U 44565559 IC50 = 199.99 nM T97747 CXN35S 44565673 IC50 = 0.3999 nM T97747 C4ZMI3 44565674 IC50 = 3.6 nM T97747 CQ8CR4 44565718 IC50 = 0.8995 nM T97747 CUB24L 44565719 IC50 = 0.7998 nM T97747 CYK2S8 44565720 IC50 = 0.2999 nM T97747 CRN02H 44565721 IC50 = 3.7 nM T97747 C7IET0 44565742 IC50 = 0.5 nM T97747 CP4J3U 44565761 IC50 = 0.57 nM T97747 CKS65Z 44565762 IC50 = 0.5998 nM T97747 C3ZRO8 44565791 IC50 = 2.999 nM T97747 CIEU13 44565852 IC50 = 0.8892 nM T97747 C6R4PT 44565853 IC50 = 0.7603 nM T97747 CIS5B7 44565854 IC50 = 1 nM T97747 CYP76Z 44565874 IC50 = 13 nM T97747 CH0V8X 44568898 IC50 > 3162.28 nM T97747 CIZ10G 44570177 IC50 = 35 nM T97747 CZ65FC 44570267 IC50 = 19 nM T97747 CBHU64 44570268 IC50 = 37 nM T97747 CY5PT0 44570269 IC50 = 30 nM T97747 C8ZA1H 44570270 IC50 = 76 nM T97747 CFH4B9 44570307 IC50 = 104 nM T97747 C4XR6K 44573097 IC50 = 320 nM T97747 C9QV3T 44573098 IC50 = 129 nM T97747 CT2BF3 44573127 IC50 = 74 nM T97747 CSD69K 44573252 IC50 = 13 nM T97747 C24BDO 44573253 IC50 = 3 nM T97747 CP6S9W 44573254 IC50 = 4 nM T97747 C6V8OC 44573255 IC50 = 7 nM T97747 CA43WF 44573256 IC50 = 6 nM T97747 C3YHW1 44573297 IC50 = 21 nM T97747 C3P8EI 44573298 IC50 = 24 nM T97747 CS01PW 44573299 IC50 = 18 nM T97747 CC38YB 44573300 IC50 = 23 nM T97747 CL7KF4 44573301 IC50 = 13 nM T97747 C3H6AO 44573302 IC50 = 40 nM T97747 CS4AC6 44573335 IC50 = 11 nM T97747 CDI9P0 44573336 IC50 = 5 nM T97747 CA0P3K 44573337 IC50 = 7 nM T97747 CT9R5H 44573338 IC50 = 4 nM T97747 CQBA10 44573339 IC50 = 23 nM T97747 CH6Q4S 44573340 IC50 = 5 nM T97747 C03RHO 44573341 IC50 = 13 nM T97747 CIXC68 44590222 IC50 = 2490 nM T97747 CU71HW 44590230 IC50 = 37.5 nM T97747 C2HUS5 44590332 IC50 = 145 nM T97747 CGM7H6 44590394 IC50 = 1 nM T97747 CJ95XB 44590395 IC50 = 1230 nM T97747 CE5U9X 44590439 IC50 = 3 nM T97747 C81IGZ 44590440 IC50 = 0.5 nM T97747 C92IJZ 44590441 IC50 = 5800 nM T97747 CI1OX6 44590557 IC50 = 7.5 nM T97747 CS8ZR6 44590583 IC50 = 14 nM T97747 CR4K7Y 44590584 IC50 = 48 nM T97747 C6ZX0E 44590585 IC50 = 5 nM T97747 C4UR9F 44590586 IC50 = 0.05 nM T97747 CDR4P2 44590633 IC50 = 0.34 nM T97747 CWEQ65 44590634 IC50 = 0.48 nM T97747 CRE37W 44590635 IC50 = 0.94 nM T97747 CCBA38 44590681 IC50 = 0.07 nM T97747 C87MFS 44590682 IC50 = 1.54 nM T97747 C24KEF 44590683 IC50 = 2.33 nM T97747 C9QSX8 44590684 IC50 = 3.76 nM T97747 C9PC7J 44590704 IC50 = 24 nM T97747 CQ6SI3 44590717 IC50 = 13.4 nM T97747 C1PV5A 44590718 IC50 = 17.9 nM T97747 CU40QM 44590719 IC50 > 25000 nM T97747 C37QZC 44590720 IC50 = 0.003 nM T97747 CB32OD 44590738 IC50 = 313 nM T97747 CUQ63O 44590739 IC50 = 41 nM T97747 CDOP14 44590750 IC50 = 0.16 nM T97747 CRDP72 44590751 IC50 = 6430 nM T97747 CTLW28 44590752 IC50 = 3.16 nM T97747 CT92AQ 44590753 IC50 = 3.4 nM T97747 C3P7HB 44590798 IC50 = 3.63 nM T97747 CZ0C5N 44590799 IC50 = 4.83 nM T97747 CBAK64 44590800 IC50 = 25.3 nM T97747 C2L6AI 44590801 IC50 = 33.7 nM T97747 C9BPW4 44590849 IC50 = 102 nM T97747 CRQ09H 44590850 IC50 = 56 nM T97747 CPV4L8 44590862 IC50 = 64.4 nM T97747 CA79TX 44590863 IC50 = 73.5 nM T97747 CIH56J 44590864 IC50 = 2310 nM T97747 CZ5HT9 44590865 IC50 = 382 nM T97747 CAC12Y 44590943 IC50 = 540 nM T97747 C2EB4O 44590944 IC50 = 1849 nM T97747 CFE24S 44590945 IC50 = 21.4 nM T97747 CHQM54 44590946 IC50 = 94.6 nM T97747 C4N1MT 46191232 IC50 = 2 nM T97747 C1SAG3 46191233 IC50 < 0.3 nM T97747 CK3N1G 46206137 IC50 > 10000 nM T97747 CV2G0F 46225342 IC50 > 2500 nM T97747 C6V9JA 46225343 IC50 = 102 nM T97747 CSET80 46225344 IC50 = 59 nM T97747 CSX9I8 46225345 IC50 = 339 nM T97747 C5G3NW 46225346 IC50 = 167 nM T97747 C28WID 46225347 IC50 = 37 nM T97747 CZFT40 46225348 IC50 = 361 nM T97747 CIA1T4 46225349 IC50 = 46 nM T97747 CS4T3F 46225350 IC50 = 28 nM T97747 C2POI6 46225394 IC50 = 65 nM T97747 C6VCG0 46225395 IC50 = 55 nM T97747 CJ9R1Y 46225428 IC50 = 1943 nM T97747 C2E6PS 46225429 IC50 = 69 nM T97747 C1G8IP 46225512 IC50 = 27 nM T97747 CW8RZ6 46225513 IC50 = 56 nM T97747 CS1H4X 46225514 IC50 = 27 nM T97747 C3H6PF 46225515 IC50 = 10 nM T97747 CZL79B 46225526 IC50 = 30 nM T97747 CK56CR 46225527 IC50 = 38 nM T97747 CQJM47 46225528 IC50 = 5 nM T97747 CVX2D6 46225529 IC50 = 66 nM T97747 C6Q2ML 46225530 IC50 = 15 nM T97747 CC9J8S 46225531 IC50 = 53 nM T97747 CV2SG0 46225532 IC50 = 1 nM T97747 CIV7G4 46225533 IC50 = 3 nM T97747 CMA4Y5 46226118 IC50 = 10000 nM T97747 C1Z3BR 46226120 IC50 = 170 nM T97747 C09LCK 46226122 IC50 = 86 nM T97747 CX6PK2 46226124 IC50 = 79 nM T97747 CAF2T0 46226126 IC50 = 130 nM T97747 CB8Q4K 46226128 IC50 = 42 nM T97747 CP10VT 46226130 IC50 = 92 nM T97747 CF85BE 46226132 IC50 = 13 nM T97747 C3YQ7A 46837425 IC50 = 10000 nM T97747 C8K4CT 46837428 IC50 > 10000 nM T97747 C8VZ9P 46837429 IC50 > 10000 nM T97747 CAG58V 46837553 IC50 = 253 nM T97747 C2E4CD 46837554 IC50 = 10000 nM T97747 CPC64Z 46837555 IC50 > 10000 nM T97747 C7XG1V 46837556 IC50 > 10000 nM T97747 C0RF1D 46864993 IC50 = 18 nM T97747 COY59E 46866599 IC50 = 8 nM T97747 CHQI42 46880774 IC50 = 6 nM T97747 CEKG54 46880775 IC50 = 30 nM T97747 CTC2X7 46880847 IC50 = 38 nM T97747 CUG39Q 46880848 IC50 = 7 nM T97747 CH0M1Q 46880849 IC50 = 5 nM T97747 CEY3D2 46880850 IC50 = 13 nM T97747 C69OGT 46880887 IC50 = 5 nM T97747 C6TN7S 46882070 IC50 > 500 nM T97747 C1YG5B 46882071 IC50 > 500 nM T97747 C23WRH 46882072 IC50 > 500 nM T97747 CLA67N 46882073 IC50 = 92 nM T97747 C9AR5O 46882074 IC50 = 98 nM T97747 C1Z8YT 46882075 IC50 = 45 nM T97747 CYV6Z5 46882076 IC50 = 14 nM T97747 C8EV6W 46882077 IC50 = 15 nM T97747 C3SJ0I 46882078 IC50 = 25 nM T97747 C5AQ1Y 46882079 IC50 = 61 nM T97747 C6XOK3 46882080 IC50 = 44 nM T97747 CUNP07 46882081 IC50 = 34 nM T97747 CSH9R7 46882082 IC50 = 23 nM T97747 C2SZI3 46882083 IC50 = 27 nM T97747 C1K3TC 46882871 IC50 = 100 nM T97747 CC9VR6 46882872 IC50 = 18 nM T97747 CXEO65 46882873 IC50 = 24 nM T97747 C69SIF 46882916 IC50 = 10 nM T97747 CMP29J 46882947 IC50 = 7 nM T97747 C20IML 46882948 IC50 = 58 nM T97747 C2U9EO 46882985 IC50 = 100 nM T97747 C18KLW 46883025 IC50 = 61 nM T97747 C8I9ZQ 46883026 IC50 = 80 nM T97747 CO8Y6D 46883027 IC50 = 24 nM T97747 C7TO8G 46883028 IC50 = 22 nM T97747 CZ6CK2 46883029 IC50 = 12 nM T97747 CU32SF 46883030 IC50 = 97 nM T97747 CM9UG5 46883031 IC50 = 10 nM T97747 CG7OL0 46883507 IC50 = 51 nM T97747 CV14GK 46888453 IC50 = 6 nM T97747 CP45CJ 46888454 IC50 = 15 nM T97747 CC7KQ1 46888455 IC50 = 11 nM T97747 CK0X4C 46888456 IC50 = 7 nM T97747 C30THG 46888478 IC50 = 3 nM T97747 CAK75S 46888479 IC50 = 4 nM T97747 C63UBP 46888480 IC50 = 8 nM T97747 CG7HE8 46888496 IC50 = 18 nM T97747 CI8MG4 46888497 IC50 = 15 nM T97747 CPO0Z8 46888498 IC50 = 465 nM T97747 CQS95E 46888499 IC50 = 9 nM T97747 CP8YH4 46888524 IC50 = 14 nM T97747 CUY17G 46888525 IC50 = 6 nM T97747 CPI6N7 46888526 IC50 = 26 nM T97747 CGZX65 46888544 IC50 = 19 nM T97747 C3NXP5 46888545 IC50 = 7 nM T97747 CM0X6G 46888546 IC50 = 44 nM T97747 C79OQJ 46888563 IC50 = 14 nM T97747 C63YJU 46888564 IC50 = 30 nM T97747 CA45RF 46888565 IC50 = 12 nM T97747 CU2TE0 46888566 IC50 = 27 nM T97747 C2PJG4 46888581 IC50 = 20 nM T97747 C5ZQ2A 46888582 IC50 = 13 nM T97747 CBD19K 46888583 IC50 = 12 nM T97747 CDI40V 46888584 IC50 = 9 nM T97747 C0FL8H 46888604 IC50 = 25 nM T97747 CVD8K7 46888605 IC50 = 30 nM T97747 C7A2BS 46888606 IC50 = 34 nM T97747 CULC94 46890340 IC50 = 26 nM T97747 CRE91L 46890341 IC50 = 62 nM T97747 CV2RH7 46890342 IC50 = 20 nM T97747 C64DLQ 46890343 IC50 = 8 nM T97747 CI9MR8 46890345 IC50 > 500 nM T97747 CWY7D6 46890346 IC50 = 33 nM T97747 C5O8EZ 46890427 IC50 = 24 nM T97747 C2KJS7 46890428 IC50 = 12 nM T97747 CJ9SL0 46890429 IC50 = 25 nM T97747 C43QJG 49768639 IC50 = 31 nM T97747 CDM18G 49768863 IC50 = 1.4 nM T97747 C3E5JT 49798079 IC50 > 30 nM T97747 CZQ54K 49798080 IC50 = 6.15 nM T97747 C32OXR 49798081 IC50 = 220.6 nM T97747 CJ5GZ2 49798082 IC50 = 1.09 nM T97747 CUQ79L 49798083 IC50 = 20.2 nM T97747 C8RVJ9 49798084 IC50 = 37.7 nM T97747 C9W7HN 49798085 IC50 = 1.71 nM T97747 C1UKV9 49798086 IC50 = 2.66 nM T97747 CFGM47 49798087 IC50 = 3.2 nM T97747 CTA1U3 49798088 IC50 = 6.15 nM T97747 CQ3R2G 49798089 IC50 = 1.62 nM T97747 CAWQ56 49798090 IC50 = 1.69 nM T97747 C61NQS 49798129 IC50 = 3.5 nM T97747 C6VPR9 49798130 IC50 = 14.6 nM T97747 C20OMQ 49798131 IC50 = 5.3 nM T97747 C72VPW 49798132 IC50 = 11 nM T97747 C4EQ0K 49798133 IC50 = 3.6 nM T97747 CV8XW0 49798156 IC50 = 17.8 nM T97747 C4I0TN 49798157 IC50 = 149.2 nM T97747 CK5S2Z 49798158 IC50 = 4 nM T97747 CQVG17 49798349 IC50 = 630.96 nM T97747 CG83TP 49798920 IC50 = 320 nM T97747 C3Y1AN 49799705 IC50 = 81 nM T97747 C7M8DB 49799707 IC50 = 57 nM T97747 CIY75R 49799711 IC50 = 42 nM T97747 CH4JV5 49864967 IC50 = 318 nM T97747 C4RQ8B 49864968 IC50 = 30 nM T97747 C8ZFG4 49864969 IC50 = 8.85 nM T97747 CZ2LD9 49864970 IC50 = 38.3 nM T97747 C7GU4O 49864971 IC50 = 1.38 nM T97747 CV4UR2 49864972 IC50 = 11.17 nM T97747 C5HKC2 49864973 IC50 = 2.98 nM T97747 C74QMJ 49864974 IC50 = 6.77 nM T97747 C5I8KJ 49864975 IC50 = 11.4 nM T97747 CP4XR3 49864976 IC50 = 30 nM T97747 C7JF3Q 49864977 IC50 = 3.98 nM T97747 CZ7CR9 50915506 IC50 = 0.4 nM T97747 CI32TR 50992246 IC50 = 5.3 nM T97747 CF0A5Z 50992494 IC50 = 0.2 nM T97747 C4IFR9 50992499 IC50 < 0.1 nM T97747 CB1VU9 50992574 IC50 = 5 nM T97747 C3S5HO 50992575 IC50 = 3 nM T97747 C51FNM 50992577 IC50 = 0.4 nM T97747 C90LTR 50992639 IC50 = 0.4 nM T97747 CWOE69 50992640 IC50 = 0.4 nM T97747 CS5C4D 50992641 IC50 = 0.3 nM T97747 CFB75J 50992642 IC50 < 0.1 nM T97747 CFG8M7 50992643 IC50 < 0.1 nM T97747 C41QJN 50992719 IC50 < 0.1 nM T97747 C4BP6M 50992720 IC50 < 0.1 nM T97747 CIO9B5 50992721 IC50 < 0.1 nM T97747 C2ST3V 50992722 IC50 < 0.1 nM T97747 C0XF6H 50993435 IC50 = 29 nM T97747 CQJ83W 50993436 IC50 = 9 nM T97747 C51DPL 50993591 IC50 = 0.1 nM T97747 C2D4XS 50993592 IC50 = 0.6 nM T97747 C70BEM 50993593 IC50 = 0.2 nM T97747 C7RX0Y 52918140 IC50 = 20 nM T97747 C7BAV4 52940989 IC50 = 41 nM T97747 C5Z1PK 52941008 IC50 = 52 nM T97747 C36JTE 52941648 IC50 = 3.3 nM T97747 CI3C8V 52942058 IC50 = 137 nM T97747 CLO38X 52942071 IC50 = 19 nM T97747 C2G1RT 52942078 IC50 = 744 nM T97747 C8V2JI 52942223 IC50 = 420 nM T97747 C9G8VW 52943283 IC50 = 99 nM T97747 CZ10FK 52943389 IC50 = 4.5 nM T97747 C03XMU 52943390 IC50 = 4.5 nM T97747 C84OYJ 52943424 IC50 = 35 nM T97747 CX3LY2 52943425 IC50 = 3100 nM T97747 CAU0O1 52943426 IC50 = 150 nM T97747 C5BEV7 52944086 IC50 = 46 nM T97747 C86MFB 52944231 IC50 = 4123 nM T97747 CQ38KM 52944537 IC50 = 11 nM T97747 C9C5OP 52944586 IC50 = 15 nM T97747 C1ZPU9 52944587 IC50 = 6.9 nM T97747 CAC4V2 52944616 IC50 = 26 nM T97747 CM24UY 52944617 IC50 = 60 nM T97747 C91GLQ 52944618 IC50 = 210 nM T97747 C64CAT 52944644 IC50 = 313 nM T97747 C4KLV6 52945332 IC50 = 34 nM T97747 CIB1K6 52945865 IC50 = 87 nM T97747 CLAH27 52946506 IC50 = 8 nM T97747 CG8S9O 52946946 IC50 > 5000 nM T97747 CA7Z6L 52946953 IC50 > 5000 nM T97747 C1C5BV 52946954 IC50 = 1.2 nM T97747 C1X9RI 52947038 IC50 = 30 nM T97747 C0F1WE 52947044 IC50 = 63 nM T97747 C8CZL6 52947063 IC50 = 22 nM T97747 C6KCU2 52947064 IC50 = 64 nM T97747 CJZK15 52947090 IC50 = 34 nM T97747 CS9UX8 52947091 IC50 = 3.7 nM T97747 CKI5X6 52947100 IC50 > 5000 nM T97747 C1ZK2O 52947741 IC50 > 5000 nM T97747 CJT61Q 52947748 IC50 = 93 nM T97747 CZK6D2 52948162 IC50 = 2819 nM T97747 C64DXZ 52948248 IC50 > 5000 nM T97747 C0ZF7V 52948264 IC50 = 8.6 nM T97747 C6LV0Q 52948295 IC50 = 20.5 nM T97747 CX2QU9 52948296 IC50 = 2.6 nM T97747 CI5EM7 52949128 IC50 = 2173 nM T97747 COH5M1 52949523 IC50 = 27 nM T97747 CU0P3Q 52949553 IC50 = 65 nM T97747 CU25FT 52949601 IC50 = 2832 nM T97747 C70QNI 53260398 IC50 = 0.3548 nM T97747 C7U1ZC 53317132 IC50 > 1000 nM T97747 C0AS8E 53318853 IC50 = 77 nM T97747 C8K5QI 53318854 IC50 = 572 nM T97747 CLP07M 53319405 IC50 = 2 nM T97747 CCV39H 53319838 IC50 = 4.6 nM T97747 CH34SY 53319839 IC50 > 1000 nM T97747 C76HPL 53321427 IC50 = 22.5 nM T97747 C1HOS5 53321482 IC50 = 312 nM T97747 CK2M9J 53321616 IC50 = 18 nM T97747 CK2JD6 53322809 IC50 = 108 nM T97747 C35XLW 53322810 IC50 = 34.8 nM T97747 C4EV2O 53323818 IC50 > 1000 nM T97747 CH3LK8 53324139 IC50 > 1000 nM T97747 COYC36 53324140 IC50 = 546 nM T97747 C48XCJ 53324141 IC50 = 206 nM T97747 CO93PA 53324304 IC50 = 23 nM T97747 CC1ER2 53324598 IC50 = 181.97 nM T97747 C9B7FY 53325088 IC50 = 211 nM T97747 C9YGA3 53325385 IC50 = 370 nM T97747 CM12CJ 53325460 IC50 = 11.1 nM T97747 CY15EU 53325639 IC50 = 26.5 nM T97747 CYA3F1 53325983 IC50 = 0.5 nM T97747 CD1SK7 53326700 IC50 = 1000 nM T97747 C8E0DF 53326701 IC50 = 204 nM T97747 C7PQ1Y 53326702 IC50 = 201 nM T97747 C8C7PV 53389082 IC50 = 4600 nM T97747 C9QD2Z 53389084 IC50 = 10010 nM T97747 CC8ME1 53389637 IC50 = 275.42 nM T97747 C13SIB 53389710 IC50 = 512.86 nM T97747 CXW05M 53389845 IC50 = 575.44 nM T97747 CS0Q8N 53389902 IC50 = 213.8 nM T97747 C4OL5J 54580080 IC50 = 2238.72 nM T97747 CL4N5M 54580081 IC50 = 19.95 nM T97747 C0O5LX 54580082 IC50 = 251.19 nM T97747 CFEK69 54580093 IC50 = 177.83 nM T97747 CRV8T5 54580467 IC50 = 40 nM T97747 C8RK1D 54580468 IC50 = 120 nM T97747 CTO38W 54580469 IC50 = 220 nM T97747 CIW93N 54581068 IC50 = 2511.89 nM T97747 CI93ZC 54581069 IC50 > 3162.28 nM T97747 CS3PM2 54581070 IC50 = 1584.89 nM T97747 C80DUA 54581071 IC50 = 1995.26 nM T97747 C05GIL 54581076 IC50 = 17.78 nM T97747 C8VQU5 54581478 IC50 = 12250 nM T97747 CU8N4Z 54581479 IC50 = 30 nM T97747 C9X4EW 54581480 IC50 = 140 nM T97747 C2AVP1 54582104 IC50 = 257.04 nM T97747 C8SEU2 54582105 IC50 = 10 nM T97747 CX0WM5 54582110 IC50 = 15.85 nM T97747 CUWR02 54583048 IC50 > 3162.28 nM T97747 CCO15Z 54583049 IC50 = 1778.28 nM T97747 CML64U 54583458 IC50 = 290 nM T97747 C6H4BZ 54583459 IC50 = 21370 nM T97747 CCRX35 54583460 IC50 = 30 nM T97747 C49QZJ 54583462 IC50 = 3800 nM T97747 CEAG79 54584051 IC50 > 3162.28 nM T97747 C53YSX 54584052 IC50 = 398.11 nM T97747 CS2UN4 54584053 IC50 = 100 nM T97747 C96PFQ 54584058 IC50 = 31.62 nM T97747 C7CAN9 54584059 IC50 = 5.012 nM T97747 C5NRH1 54584427 IC50 = 970 nM T97747 CTRG70 54585004 IC50 > 3162.28 nM T97747 CHPB98 54585369 IC50 = 1760 nM T97747 CP8Q6M 54585383 IC50 = 5620 nM T97747 CH7NT9 54585384 IC50 = 130 nM T97747 CI1U4V 54585385 IC50 = 3390 nM T97747 C9ONK2 54585963 IC50 = 251.19 nM T97747 CQP1B8 54585964 IC50 = 8.913 nM T97747 CB82XJ 54585972 IC50 > 3162.28 nM T97747 CGS76T 54586286 IC50 = 180 nM T97747 CW97CT 54586339 IC50 = 100 nM T97747 CEA41I 54587374 IC50 = 17010 nM T97747 C7PHF2 54752872 IC50 = 10100 nM T97747 CVA1S8 54752874 IC50 = 9200 nM T97747 CG4U7M 54753646 IC50 = 5400 nM T97747 CM0Z8W 56647023 IC50 = 6.9 nM T97747 CYR89T 56647076 IC50 = 6.4 nM T97747 C57DEP 56657984 IC50 = 59000 nM T97747 CWF8C3 56657986 IC50 = 180000 nM T97747 C1K5GS 56659271 IC50 = 48090 nM T97747 CGK57R 56661522 IC50 = 81000 nM T97747 CMV8C3 56661524 IC50 = 25000 nM T97747 CZN3H8 56661526 IC50 = 20000 nM T97747 C2BMX7 56661530 IC50 = 1148000 nM T97747 C48GTM 56664935 IC50 = 50000 nM T97747 CKQG84 56664937 IC50 = 23000 nM T97747 CA9ML1 56664939 IC50 = 190000 nM T97747 CFYI08 56668364 IC50 = 270000 nM T97747 C4TXR2 56669615 IC50 = 7800 nM T97747 CJC18T 56671869 IC50 = 120000 nM T97747 CNX6F5 56673133 IC50 = 15240 nM T97747 CXI8E3 56675256 IC50 = 140000 nM T97747 C5U1RV 56676454 IC50 = 37610 nM T97747 CGS0W3 56678574 IC50 = 23000 nM T97747 CGS5P2 56678576 IC50 = 21000 nM T97747 CUL60G 56678578 IC50 = 35000 nM T97747 C5LJ8C 56681915 IC50 = 5200 nM T97747 COS02D 56681917 IC50 = 3900 nM T97747 C3A7OC 56683102 IC50 = 8400 nM T97747 CHM6Z8 56750906 IC50 = 36000 nM T97747 CQ9S6H 56754672 IC50 = 70000 nM T97747 C97HKS 57331246 IC50 > 1000 nM T97747 CR3HF8 57331274 IC50 = 25.73 nM T97747 CXV90D 57331275 IC50 = 76.03 nM T97747 CFC2Q4 57331276 IC50 = 35.47 nM T97747 C50UMI 57331277 IC50 = 320.33 nM T97747 C9Y6MI 57331278 IC50 = 25.53 nM T97747 CVDQ59 57331304 IC50 = 64.07 nM T97747 C6VUQ9 57331305 IC50 = 525 nM T97747 C36BJH 57331306 IC50 = 93.53 nM T97747 CV7X0G 57331307 IC50 = 26.37 nM T97747 CX58OH 57331308 IC50 = 473.33 nM T97747 C5JFZ1 57331339 IC50 = 75.3 nM T97747 CXO80S 57331340 IC50 = 202.43 nM T97747 CNS7H5 57335017 IC50 = 7300 nM T97747 CBF53W 57384005 IC50 = 0.3 nM T97747 CF1OM2 57384006 IC50 = 0.3 nM T97747 C16ZHL 57390535 IC50 = 8 nM T97747 CZOY39 57391591 IC50 = 810 nM T97747 CCA7D3 57391720 IC50 = 8.9 nM T97747 C5ND1L 57391721 IC50 = 0.44 nM T97747 C5QD2I 57391722 IC50 = 0.55 nM T97747 CCKJ07 57392302 IC50 = 387 nM T97747 C0YX7L 57392303 IC50 = 0.7 nM T97747 CK59VA 57392726 IC50 = 2850 nM T97747 CPQC75 57393451 IC50 = 3.5 nM T97747 CO29JI 57394057 IC50 = 1.6 nM T97747 C3F4XE 57394058 IC50 = 7 nM T97747 CGV90O 57395178 IC50 = 3.1 nM T97747 C9G6OJ 57395179 IC50 = 5 nM T97747 CGR9F3 57395184 IC50 < 0.1 nM T97747 CSH0P9 57395816 IC50 = 12.3 nM T97747 C3AB8V 57395817 IC50 = 1.5 nM T97747 C23QVB 57395818 IC50 = 130 nM T97747 CVXD20 57396843 IC50 = 5.4 nM T97747 C75SYT 57396949 IC50 = 229 nM T97747 CWU1I0 57396950 IC50 < 0.1 nM T97747 CR41GU 57396951 IC50 = 3700 nM T97747 C9YT0S 57396952 IC50 = 0.69 nM T97747 CTH3P5 57396953 IC50 < 0.1 nM T97747 C0R1ET 57397595 IC50 = 116 nM T97747 C23IKA 57397596 IC50 = 11 nM T97747 CZ29HN 57397597 IC50 = 3 nM T97747 CC72RQ 57397598 IC50 = 2.4 nM T97747 CH58PW 57397603 IC50 = 1586 nM T97747 CA2IY7 57398009 IC50 = 1300 nM T97747 CK97BJ 57400372 IC50 = 39 nM T97747 C19SNT 57400373 IC50 = 162 nM T97747 CA5KO3 57400374 IC50 = 1.1 nM T97747 CT31JR 57400375 IC50 = 794 nM T97747 C0H7ME 57401041 IC50 = 90 nM T97747 CCJ1I2 57401042 IC50 = 12 nM T97747 C5NDS6 57402175 IC50 = 1.6 nM T97747 CRUX38 57402798 IC50 = 50 nM T97747 CV96NF 57402799 IC50 = 3 nM T97747 C9ER8K 57402800 IC50 = 2 nM T97747 C37NBY 57402801 IC50 = 0.09 nM T97747 CA7TX2 57402802 IC50 = 0.98 nM T97747 CXYB90 57403173 IC50 = 1000 nM T97747 CU4S6M 57403931 IC50 = 15 nM T97747 CC0D8X 57403932 IC50 = 0.68 nM T97747 CHJ87A 57656833 IC50 = 22 nM T97747 CZ71SN 58282592 IC50 = 650 nM T97747 C0YWT1 58509213 IC50 > 10000 nM T97747 C6JKM0 58834906 IC50 = 0.6 nM T97747 CR8L7P 58834946 IC50 = 0.9 nM T97747 CF9Z0L 58834953 IC50 = 1.1 nM T97747 CMJ59Z 58834969 IC50 = 0.4 nM T97747 CM6Z7S 58835000 IC50 = 1.3 nM T97747 C4PWA9 58835024 IC50 = 1.4 nM T97747 C7RXU8 58835027 IC50 = 1.3 nM T97747 CC36OU 58835113 IC50 = 0.9 nM T97747 C2XRL5 58835114 IC50 = 1.1 nM T97747 CN3RD2 58835155 IC50 = 1.5 nM T97747 CCR4T7 58835217 IC50 = 0.7 nM T97747 C76HQB 59458061 IC50 = 0.4 nM T97747 C5KUQ8 59458103 IC50 = 1.7 nM T97747 CEI9H7 59458159 IC50 = 8.6 nM T97747 CQTK25 59458213 IC50 = 5.3 nM T97747 C46UHJ 59458228 IC50 = 0.4 nM T97747 C7SOK2 59458245 IC50 = 1 nM T97747 C27NIL 59458247 IC50 = 0.9 nM T97747 C6GPD8 59959034 IC50 = 1 nM T97747 CT0NG6 62706106 IC50 = 0.7 nM T97747 CKA9V2 62706107 IC50 = 0.11 nM T97747 CB91CU 62706108 IC50 = 0.9 nM T97747 CG58WC 62706109 IC50 = 0.8 nM T97747 CA4RU3 62706110 IC50 = 0.3 nM T97747 C0N8XJ 62707281 IC50 = 9200 nM T97747 CHU5Q0 62707283 IC50 = 16300 nM T97747 CJ2S6W 62707285 IC50 > 100000 nM T97747 CTC5D7 62707286 IC50 > 30000 nM T97747 C9NGJ8 62707287 IC50 = 6500 nM T97747 C40ORM 62707443 IC50 = 7800 nM T97747 CX4MO7 62707444 IC50 = 10000 nM T97747 CF4X6H 62707445 IC50 = 8400 nM T97747 CPDZ56 62707446 IC50 = 4600 nM T97747 C2N9YG 62707447 IC50 = 48100 nM T97747 C3X8YK 62707448 IC50 = 15200 nM T97747 CAY3H7 62707598 IC50 = 37600 nM T97747 CQR25M 66767933 IC50 = 321 nM T97747 CO62SG 66768099 IC50 = 137 nM T97747 CC81NU 66768640 IC50 = 1242 nM T97747 CCB1T5 68764898 IC50 = 2.4 nM T97747 C5O0JN 68764925 IC50 = 3 nM T97747 C70QJS 68767049 IC50 = 3.4 nM T97747 C8VU1C 68767078 IC50 = 22 nM T97747 C2YRL3 68769802 IC50 = 18 nM T97747 C39SPK 68772423 IC50 = 190 nM T97747 CV8E4C 69696607 IC50 = 750000 nM T97747 CDF0Q5 69697526 IC50 = 640000 nM T97747 C0POJ4 70685193 IC50 = 400 nM T97747 CU62NM 70688699 IC50 = 16400 nM T97747 CQOD53 70690765 IC50 = 10500 nM T97747 CZ0Y7T 70692897 IC50 > 30000 nM T97747 C1ACG8 70692902 IC50 = 9200 nM T97747 CW6UA5 70694934 IC50 > 30000 nM T97747 CV10AS 70694935 IC50 > 30000 nM T97747 CV53PW 70694941 IC50 = 13700 nM T97747 CW0B9M 71451541 IC50 = 31.1 nM T97747 C0F7NL 71451877 IC50 = 0.17 nM T97747 CDJN04 71458736 IC50 = 1.2 nM T97747 CP2UK0 71458737 IC50 = 14.3 nM T97747 CIP7D8 71462570 Ki = 1 nM T97747 CI8Q1K 71717723 Ki = 31 nM T97747 CP5NQ2 71718331 Ki = 210 nM T97747 CZ5C6V 71718930 Ki = 150 nM T97747 CC8JQ9 71719547 Ki = 50 nM T97747 C8CB3S 72711047 IC50 = 2.5 nM T97747 CIV83U 72711048 IC50 = 15 nM T97747 CFY8W4 72711049 IC50 = 34.8 nM T97747 CZG4V5 72711050 IC50 = 157.6 nM T97747 C8E2FK 72711051 IC50 = 700.8 nM T97747 CA5B9Z 72711277 IC50 = 4.7 nM T97747 C4UJW6 72711278 IC50 = 7.1 nM T97747 CGT0X3 72711279 IC50 = 832 nM T97747 CZI06T 72711280 IC50 = 300.7 nM T97747 C7XS9L 72711281 IC50 = 117.1 nM T97747 CM0OT6 72711506 IC50 = 24.7 nM T97747 C4HG7X 72711507 IC50 = 6.4 nM T97747 CTG02P 72711508 IC50 = 3.6 nM T97747 C37CFT 72711739 IC50 = 0.9 nM T97747 C7Q6PX 72711740 IC50 = 0.8 nM T97747 C8BG4M 72711741 IC50 = 0.9 nM T97747 C86FZB 72711742 IC50 = 1.2 nM T97747 CI0ZP4 72711955 IC50 = 5.9 nM T97747 CKR7P1 72711956 IC50 = 1.2 nM T97747 CHR42S 72711958 IC50 = 0.8 nM T97747 CMUB57 72712158 IC50 = 56 nM T97747 C6ISW8 72712159 IC50 = 12.4 nM T97747 C95SNW 72712160 IC50 = 169 nM T97747 CFAM28 72712161 IC50 = 17.9 nM T97747 C4MN3V 72712371 IC50 = 43.5 nM T97747 C6HR8T 72712372 IC50 = 279.5 nM T97747 C4Q2FZ 72712373 IC50 = 15.2 nM T97747 CT30UZ 72712374 IC50 = 50.7 nM T97747 C4ZSH1 72712375 IC50 > 1000 nM T97747 C9BK3P 72712597 IC50 = 15.8 nM T97747 C4ZFJ9 72712598 IC50 = 0.3 nM T97747 C0L2NB 72713858 IC50 = 39 nM T97747 C5VP8L 72713859 IC50 = 65.7 nM T97747 C1PO6A 72713860 IC50 = 13.6 nM T97747 CQ27VU 72713861 IC50 = 9039 nM T97747 CUI40C 72714076 IC50 = 14 nM T97747 C4ZRE2 72714077 IC50 = 1465 nM T97747 C4G1OR 72714078 IC50 = 1.2 nM T97747 C3Z7NO 72714079 IC50 = 1.5 nM T97747 CLA8B7 72714317 IC50 = 1702 nM T97747 C5MOY1 72714318 IC50 = 91 nM T97747 C9KB5E 72714319 IC50 = 195 nM T97747 CWY19V 72714320 IC50 = 11.7 nM T97747 C9XOJ0 72714321 IC50 = 10.4 nM T97747 CSV58N 73345281 Ki = 30000 nM T97747 CXD8A1 73346388 IC50 = 9.6 nM T97747 C82YDH 73346389 IC50 = 7.5 nM T97747 CNPK53 73346454 IC50 = 70800 nM T97747 CM19JQ 73346460 IC50 = 115000 nM T97747 C5XW1B 73346461 IC50 = 61000 nM T97747 CUQ94P 73346462 IC50 = 47000 nM T97747 CCJ01L 73347894 IC50 = 3.4 nM T97747 C6LTC1 73347956 IC50 = 77000 nM T97747 CMK7G0 73347961 IC50 = 63000 nM T97747 CR54VT 73349498 IC50 = 45000 nM T97747 C2TN1Z 73349499 IC50 = 65700 nM T97747 CA3X1K 73349500 IC50 = 88100 nM T97747 C4UP2I 73349506 IC50 = 56000 nM T97747 CO7ZS8 73349882 Ki = 5100 nM T97747 C1RV2N 73351054 IC50 = 138000 nM T97747 CFH03E 73351055 IC50 = 90000 nM T97747 CZ4C1R 73351059 IC50 = 28000 nM T97747 CFC9T7 73351060 IC50 = 51800 nM T97747 CD20KR 73352463 IC50 = 12.7 nM T97747 COGK67 73352528 IC50 = 92200 nM T97747 C04HGN 73352529 IC50 = 61000 nM T97747 C4D1TK 73352534 IC50 = 59000 nM T97747 CZWL45 73353307 EC50 = 0.18 nM T97747 C1MK9E 73354018 IC50 = 66200 nM T97747 C9TQ1F 73355478 IC50 = 22.5 nM T97747 CHKD46 73355549 IC50 = 77800 nM T97747 C2G5NZ 73355550 IC50 = 28700 nM T97747 C98NGO 73355552 IC50 = 73000 nM T97747 C0O3UA 73355553 IC50 = 38800 nM T97747 C9URF8 73355554 IC50 = 43500 nM T97747 C84QWC 73357100 IC50 = 64000 nM T97747 C8PJU5 76308345 IC50 = 599.79 nM T97747 CJPW31 76308985 IC50 = 1499.68 nM T97747 C82LXO 76308986 IC50 = 34.99 nM T97747 CV73GF 76309037 IC50 = 100 nM T97747 CHEU38 76310164 IC50 = 86.7 nM T97747 C3W7VP 76310165 IC50 = 151.8 nM T97747 C6JAT5 76311990 IC50 = 399.94 nM T97747 C58AGV 76312665 IC50 = 209.89 nM T97747 C5J6YC 76312666 IC50 = 57.02 nM T97747 C7WO1R 76313867 IC50 = 251.67 nM T97747 COZM91 76315543 IC50 = 1000 nM T97747 CF20LV 76315544 IC50 = 6998.42 nM T97747 C1EV0K 76316185 IC50 = 10.99 nM T97747 CS3BE1 76316241 IC50 = 1.995 nM T97747 CA72FV 76316242 IC50 = 39.81 nM T97747 CZ6L7V 76316949 IC50 = 14.4 nM T97747 C3QU8F 76317388 IC50 = 125.81 nM T97747 C20DSV 76317476 IC50 = 27 nM T97747 C24QYM 76317477 IC50 > 1000 nM T97747 C5TW0Z 76319890 IC50 = 169.82 nM T97747 CRN39I 76319891 IC50 = 3698.28 nM T97747 CHJ74V 76319944 IC50 = 1000 nM T97747 C9TEP7 76321110 IC50 > 1000 nM T97747 C9IZV4 76321206 IC50 = 3 nM T97747 C7QA1M 76322864 IC50 = 1000 nM T97747 CI97JM 76323541 IC50 = 1399.59 nM T97747 CTW39E 76324825 IC50 = 2.6 nM T97747 CL92XF 76324826 IC50 = 360 nM T97747 CH60RK 76327118 IC50 = 839.46 nM T97747 CL5Y7P 76327119 IC50 = 599.79 nM T97747 CFY46V 76327120 IC50 = 100 nM T97747 CG81BM 76327166 IC50 = 0.7943 nM T97747 CPR37U 76327885 IC50 = 112 nM T97747 CPV7L2 76330768 IC50 = 449.78 nM T97747 CLJ7E0 76330769 IC50 = 319.89 nM T97747 CFR3L2 76330770 IC50 = 46.99 nM T97747 CFLJ46 76330829 IC50 = 0.7586 nM T97747 CKA2Z8 76334365 IC50 = 1000 nM T97747 C8DW4B 76335572 IC50 = 196.9 nM T97747 C8ENW7 76335673 IC50 = 0.96 nM T97747 C03MUJ 86294766 IC50 = 48000 nM T97747 CI67KS 89702731 IC50 = 126 nM T97747 CH58FP 90656325 IC50 = 10300 nM T97747 C89GMZ 90656326 IC50 = 6450 nM T97747 CRFE08 90656327 IC50 > 50000 nM T97747 CV1DY8 90656328 IC50 = 16800 nM T97747 C5UW7K 90656329 IC50 > 50000 nM T97747 CZN8T2 90656330 IC50 = 6290 nM T97747 C7B2PH 90656331 IC50 > 50000 nM T97747 CPY6G0 90656332 IC50 > 50000 nM T97747 CPZ46K 90656333 IC50 = 23000 nM T97747 CAYE46 90656334 IC50 = 9800 nM T97747 C0KCP6 90656335 IC50 = 41200 nM T97747 C37ZBS 90656336 IC50 > 50000 nM T97747 CP5X4Y 90656337 IC50 = 45800 nM T97747 CEH42L 90656338 IC50 = 45900 nM T97747 CYX8F5 90656339 IC50 = 27000 nM T97747 C21GTQ 90656340 IC50 = 19800 nM T97747 C2NWY9 90656341 IC50 = 5100 nM T97747 CQ95YH 90656342 IC50 = 25600 nM T97747 C0LYS7 90656343 IC50 = 28100 nM T97747 C24AMG 90664936 IC50 = 35 nM T97747 CY8E3J 90665058 IC50 = 21 nM T97747 CYP01O 90665176 IC50 = 71 nM T97747 CJ2ME7 90666577 IC50 = 622 nM T97747 CEA06F 90666578 IC50 = 14.2 nM T97747 CIY0P6 90666579 IC50 = 1570 nM T97747 CI53XQ 90666580 IC50 = 7910 nM T97747 C3L6KU 91820689 IC50 = 3 nM T97747 C6ENV5 100951623 EC50 > 10000 nM T97747 CFRK67 118727171 IC50 = 8.3 nM T97747 C0LC6G 118727172 IC50 = 15.1 nM T97747 CIY59U 118727173 IC50 = 25.1 nM T97747 CL4H7J 118727174 IC50 = 6.6 nM T97747 C53EMI 118727175 IC50 = 30.1 nM T97747 C6J4DP 118727176 IC50 = 11.7 nM T97747 CYR91T 118727177 IC50 = 319.9 nM T97747 CZ20TS 118727178 IC50 = 25.1 nM T97747 C68DNS 118727179 IC50 = 30 nM T97747 CM67QT 118727180 IC50 = 10.9 nM T97747 CV1R5P 118727181 IC50 = 2158 nM T97747 C45PVA 118727182 IC50 = 204.1 nM T97747 C5KJW2 118727183 IC50 = 259.7 nM T97747 C03FHC 118727184 IC50 = 17.1 nM T97747 CGW9I8 118727185 IC50 = 33.2 nM T97747 CP57BR 118727186 IC50 = 8.8 nM T97747 CV5MD3 118727187 IC50 = 906 nM T97747 CJO04D 118727188 IC50 = 49.9 nM T97747 C8F6AV 118727189 IC50 = 3 nM T97747 C16VCE 118727190 IC50 = 239.5 nM T97747 C4E7QF 118727191 IC50 = 163.8 nM T97747 CXM94Y 118727192 IC50 = 6290 nM T97747 C5L3SI 122185608 IC50 = 12700 nM T97747 CQ5WN1 122185610 IC50 = 17300 nM T97747 CSR65M 122185612 IC50 = 12900 nM T97747 CWG5Y3 122185614 IC50 = 30100 nM T97747 CWV1B6 122185616 IC50 = 26800 nM T97747 C9FND3 122185618 IC50 = 38500 nM T97747 CV8H0G 122185620 IC50 = 46200 nM T97747 C57TSL 122185622 IC50 = 121500 nM T97747 C1XDO2 122185624 IC50 = 67700 nM T97747 C6X1JP 122185626 IC50 = 80900 nM T97747 CR3MI5 122185628 IC50 = 101200 nM T97747 CEL59A 122185630 IC50 = 173900 nM T97747 C0Z4RT 122185632 IC50 = 19300 nM T97747 C5L7KA 122185634 IC50 = 69000 nM T97747 CK67LU 122185636 IC50 = 23900 nM T97747 C2G7TC 122185638 IC50 = 18700 nM T97747 CD1MG8 122185640 IC50 = 1350 nM T97747 C60LPW 122668161 IC50 = 51.7 nM T97747 C4KQS3 122668167 IC50 = 33 nM T97747 C85JKN 122668190 IC50 = 3.1 nM T97747 C5DUQ7 122668213 IC50 = 2.6 nM T97747 C8T9ON 126567253 IC50 = 15.8 nM T97747 CTAG09 126567264 IC50 = 2.8 nM T97747 CFWG31 126567273 IC50 = 82.6 nM T97747 CN68LA 126567277 IC50 = 12 nM T97747 CK36LH 126567281 IC50 = 27.1 nM T97747 CUFI59 126567286 IC50 = 6.8 nM T97747 C5QT4N 126567306 IC50 = 9.1 nM T97747 CK73PJ 129907953 EC50 = 42460 nM T97747 CS4M1X 129908109 EC50 = 29670 nM T97747 C8QYG0 129908110 EC50 = 11220 nM T97747 CGD5O4 129908111 EC50 = 18850 nM T97747 C0PH6K 129908112 EC50 > 50000 nM T97747 C7WXL1 129908179 EC50 > 50000 nM T97747 C8P9OC 129908195 EC50 = 15990 nM T97747 CNC2W3 129908196 EC50 = 22840 nM T97747 C14IAU 129908213 EC50 > 50000 nM T97747 CE80MX 129908214 EC50 > 50000 nM T97747 C6N0SF 129908215 EC50 > 50000 nM T97747 CG1M2A 129908240 EC50 > 50000 nM T97747 CJS4A1 129908281 EC50 = 4850 nM T97747 C2QSU0 129908301 EC50 = 16250 nM T97747 C2U4JE 129908428 EC50 = 16560 nM T97747 CV72QT 129908452 EC50 = 16830 nM T97747 CAX21P 129908453 EC50 = 18770 nM T97747 CSG86U 129908454 EC50 = 23140 nM T97747 C17ZKU 129908455 EC50 = 30630 nM T97747 CY9MZ7 129908456 EC50 = 18340 nM T97747 CONW96 129908557 EC50 > 50000 nM T97747 C2YB7V 129908558 EC50 = 36300 nM T97747 CC9S4Q 129908559 EC50 > 200000 nM T97747 C5WGK9 129908560 EC50 = 55370 nM T97747 CSD1X5 132572938 EC50 > 10 nM T97747 CV8N7E 137635442 EC50 > 10 nM T97747 C52MBZ 137638300 EC50 > 10 nM T97747 CL8P3K 137641868 EC50 > 10 nM T97747 CR2HZ3 137648323 EC50 > 10 nM T97747 C2WT5B 137654404 EC50 > 10 nM T97747 C0X5EI 137655931 EC50 > 10 nM T97747 CYV7M3 137660245 EC50 = 2470 nM T97747 C32SJE 145961982 IC50 = 660 nM T97747 C56KSZ 145967247 IC50 = 1.288 nM T97747 CXA2G0 145967391 IC50 = 1100 nM T97747 C1SQ3H 145982775 IC50 = 2.9 nM T97747 CY0S1F 145983098 IC50 = 296.4 nM T97747 CCHZ83 145983159 IC50 = 24.5 nM T97747 C87XGI 145983513 IC50 = 16.2 nM T97747 CTRV17 145983733 IC50 = 2.9 nM T97747 CVD12G 145983844 IC50 = 20.6 nM T97747 CS26EW 145984103 IC50 = 87.9 nM T97747 CQ5EN9 145984502 IC50 = 2.6 nM T97747 C2ANL3 145984591 IC50 = 4 nM T97747 C50AOD 145984717 IC50 = 5.4 nM T97747 C4HAP0 145984727 IC50 = 2.3 nM T97747 C53PGI 145984829 IC50 = 2.6 nM T97747 C5IZJ6 145985042 IC50 = 2.9 nM T97747 C6YW8A 145985237 IC50 = 8.1 nM T97747 CYG9S8 145985461 IC50 = 2.8 nM T97747 CQOR04 145985672 IC50 = 3 nM T97747 C0JOG7 145985889 IC50 = 5.2 nM T97747 C4LA2T 145985894 IC50 = 9.7 nM T97747 CB0FC5 145986021 IC50 = 2.3 nM T97747 CP2Z5X 145986145 IC50 = 4.7 nM T97747 CNC59J 145986205 IC50 = 251.6 nM T97747 CAF10K 145986277 IC50 = 6.8 nM T97747 CFN4J8 145996522 EC50 = 4.467 nM T97747 CXT09R 154572822 IC50 = 287 nM T97747 COP6C1 155491018 EC50 = 5 nM T97747 CVQ31N 155513284 IC50 = 371.54 nM T97747 C86OHR 155529593 IC50 = 3469 nM T97747 CVS37C 155531379 IC50 = 1570 nM T97747 CZ04TG 155540798 IC50 = 323.59 nM T97747 C80LBZ 155554273 IC50 = 123.03 nM T97747 D01LRC 6479877 IC50 = 5400 nM T97747 D06MBD 11176403 IC50 < 3000 nM T97747 D06QRP 5311123 Ki = 66 nM T97747 D06XIC 6480205 IC50 = 9000 nM T97747 D06XRS 4716524 IC50 = 1099.01 nM T97747 D0BD3G 11188669 IC50 = 1000 nM T97747 D0BD6A 10278617 IC50 = 5.1 nM T97747 D0E4YP 9873888 Ki = 1.4 nM T97747 D0I3IZ 11267381 IC50 = 1700 nM T97747 D0J3BT 16663418 IC50 = 3.5 nM T24587 D0B2WQ 3025944 IC50 = 9 nM T24587 CW67XG 65275 IC50 = 248000 nM T24587 C2LM0G 95802 IC50 > 1000000 nM T24587 CPF4T0 95803 IC50 = 493000 nM T24587 CNFP76 95805 IC50 > 1000000 nM T24587 C48VUD 445940 IC50 > 1000000 nM T24587 C7WS0Q 5329494 IC50 = 1006000 nM T24587 CUJ4F7 5329495 IC50 > 100000 nM T24587 C5RQ9J 5329499 IC50 > 1000000 nM T24587 CSU26A 5329500 IC50 = 11500 nM T24587 CK62GL 5329503 IC50 = 9900 nM T24587 C8ZU6I 5329504 IC50 = 16000 nM T24587 C94XIV 5329505 IC50 > 1000000 nM T24587 C0CEX8 5329506 IC50 = 37500 nM T24587 C9ZYO0 5329508 IC50 = 95000 nM T24587 C4S7QY 5329509 IC50 > 1000000 nM T24587 C2R9AY 5329510 IC50 = 200 nM T24587 C0L4FT 5329511 IC50 = 1600 nM T24587 CE5M7B 5329520 IC50 = 548000 nM T24587 CJZ15B 5329525 IC50 > 1000000 nM T24587 CSRJ03 5329526 IC50 > 1000000 nM T24587 CBC0J5 6418797 IC50 = 38 nM T24587 CGE47Q 10130617 IC50 = 170000 nM T24587 CZ76SO 10264728 IC50 = 51 nM T24587 CW58MJ 10489822 IC50 > 1000000 nM T24587 C9TFC3 10536741 IC50 = 550 nM T24587 C8KRU4 10539378 IC50 = 18000 nM T24587 C6BGP8 10586491 IC50 = 230 nM T24587 CAT01B 10587534 IC50 = 1900 nM T24587 CGI1Y9 10632766 IC50 = 93200 nM T24587 C1YWL8 10635398 IC50 > 1000000 nM T24587 CTD86L 10639059 IC50 > 1000000 nM T24587 C92BYS 10659580 IC50 > 1000000 nM T24587 COD16Q 10681258 IC50 = 554000 nM T24587 CIZA82 10684050 IC50 = 12000 nM T24587 C8D9AH 10704094 IC50 > 1000000 nM T24587 CI7G2F 10731331 IC50 = 350 nM T24587 C8EDL1 10753919 IC50 = 1600 nM T24587 CX40RF 10755107 IC50 = 2500 nM T24587 C0NR7X 24905366 IC50 = 9 nM T24587 CAD3O6 44353161 IC50 = 450 nM T24587 CLI0A1 44353224 IC50 = 3 nM T24587 CEDI38 44353255 IC50 = 32 nM T24587 CARU42 44353267 IC50 = 680 nM T24587 CBI8P9 44353279 IC50 = 25000 nM T24587 C34RQB 44353281 IC50 = 30 nM T24587 CUI60E 44353291 IC50 = 30 nM T24587 CDP2G3 44353297 IC50 = 250 nM T24587 CSFN21 44353306 IC50 = 450 nM T24587 CKTH40 44353315 IC50 = 2000 nM T24587 CXR8I4 44365980 IC50 = 1400 nM T24587 CW2ZJ8 44365981 IC50 = 120 nM T24587 CQOM16 44366006 IC50 = 60 nM T24587 C1OLX9 44366017 IC50 = 70 nM T24587 CLIN75 44366018 IC50 = 130 nM T24587 CV9O3M 44366088 IC50 = 40 nM T24587 CX65BA 44366346 IC50 = 200 nM T24587 C6LR5U 44366352 IC50 = 90 nM T24587 C8PC3K 44366360 IC50 = 220 nM T24587 C8RAH4 44366361 IC50 = 6000 nM T24587 C7O9JM 44366362 IC50 = 8500 nM T24587 CQS09X 44366363 IC50 = 80 nM T24587 CE1I4B 44366364 IC50 = 5 nM T24587 C14DXP 44366376 IC50 = 350 nM T24587 C56OHJ 44366377 IC50 = 18 nM T24587 COJ36K 44457175 IC50 = 2600 nM T24587 C0QLY2 51351517 IC50 = 1000 nM T24587 CL4TQ9 51351519 IC50 = 4700 nM T24587 CWDE94 53317586 IC50 = 19000 nM T24587 CX7SW8 53317587 IC50 > 600000 nM T24587 CK4T2C 53320184 IC50 = 20000 nM T24587 CGOF98 53321500 IC50 = 5700 nM T24587 C1PY2L 53326715 IC50 = 13000 nM T24587 C6ZR1I 53326716 IC50 > 600000 nM T24587 C56ENB 53326717 IC50 = 320 nM T24587 CV7S0I 71449867 IC50 = 25 nM T24587 C42ODZ 71462400 IC50 = 86 nM T24587 CEL16K 155523983 Ki = 24 nM T24587 D01FJB 5329512 IC50 > 1000000 nM T24587 D04RNU 181029 IC50 = 130 nM T24587 D07BTU 9860003 IC50 = 1300 nM T24587 D0B5BG 4578 IC50 = 39 nM T24587 D0R1FT 4564 IC50 > 1000000 nM T24587 D0Z8EI 179571 IC50 = 2700 nM T86364 CB59HM 11570626 IC50 = 11580 nM T86364 CWH6T3 72548703 IC50 = 0.47 nM T86364 CT4Z1R 127034614 IC50 = 11.48 nM T86364 CU12JI 127035881 IC50 = 9 nM T86364 C4AMZ8 134130418 IC50 = 0.11 nM T86364 C79AJP 145994302 IC50 = 4.9 nM T64553 D01PZD 5329098 IC50 = 20700 nM T64553 D04LVK 57379345 IC50 = 9700 nM T64553 D02NNV 3038525 IC50 > 5000 nM T64553 D02RJY 11442891 IC50 > 10000 nM T64553 D03HUX 49792852 IC50 > 10000 nM T64553 D03LWG 53235510 IC50 > 10000 nM T64553 D06KTJ 53252276 IC50 = 75 nM T64553 D07EHV 44814409 IC50 > 10000 nM T64553 D07HPJ 11476171 IC50 > 10000 nM T64553 D0A1AQ 5329099 IC50 = 28400 nM T64553 D0E3TC 44259 IC50 = 1.3 nM T64553 D0LF1U 5287969 IC50 > 50000 nM T64553 D0O0LS 25141092 IC50 > 10000 nM T64553 D0Q7RE 16007391 Ki = 8200 nM T64553 D0Q9UX 16718576 IC50 > 10000 nM T64553 D0R9IU 44462758 IC50 = 60 nM T64553 D0S5RC 3025986 IC50 > 40000 nM T64553 D0S6TK 11213558 IC50 = 42 nM T64553 D03BNU 59604787 IC50 > 10000 nM T64553 D09HEV 6539952 IC50 > 20000 nM T64553 D0T3ME 156422 IC50 > 20000 nM T64553 C6D4GE 3134 Ki > 10000 nM T64553 CBPM40 4878 IC50 > 100000000 nM T64553 C4MNG8 445840 IC50 > 10000 nM T64553 C1ZG2U 449087 IC50 > 10000 nM T64553 CHE8K4 1301845 IC50 = 29000 nM T64553 C19-AUG 1927544 IC50 = 22000 nM T64553 CY35GB 2241431 IC50 = 14000 nM T64553 CHGS79 3551941 Ki > 10000 nM T64553 CTID76 5282335 IC50 > 50000 nM T64553 CT94JS 5329138 IC50 = 25000 nM T64553 CUE64R 5329179 IC50 = 65000 nM T64553 CHA68G 5329180 IC50 = 36000 nM T64553 CNTD47 5329181 IC50 = 26000 nM T64553 CYFD81 5329182 IC50 = 94000 nM T64553 C21IKR 5329183 IC50 = 184000 nM T64553 C45ZME 5329185 IC50 = 55000 nM T64553 C5U7DB 5329186 IC50 > 500000 nM T64553 CQ6X8M 5329189 IC50 = 96000 nM T64553 C5HG9S 5329194 IC50 = 4000 nM T64553 CHV5Y6 5329195 IC50 = 5000 nM T64553 C3DOZ9 5329196 IC50 = 3000 nM T64553 CT61MB 5329197 IC50 = 3000 nM T64553 C6OT4G 5329198 IC50 = 228000 nM T64553 CROF47 5329199 IC50 = 128000 nM T64553 CHNM67 5329200 IC50 > 500000 nM T64553 C1G6ZU 5329201 IC50 = 43000 nM T64553 CA2HW9 5329202 IC50 = 32000 nM T64553 C30CUW 5329203 IC50 = 14000 nM T64553 C0UY4Q 5329204 IC50 = 11000 nM T64553 C3QIN5 5329205 IC50 = 31000 nM T64553 C5OBU1 5329206 IC50 = 7000 nM T64553 C2GKT3 5329207 IC50 = 4000 nM T64553 CKB23P 5329209 IC50 = 5000 nM T64553 CDL19N 5329212 IC50 = 3000 nM T64553 CI03PS 5329214 IC50 > 500000 nM T64553 C43NAT 5329215 IC50 = 14000 nM T64553 C9D3WP 5329216 IC50 = 8000 nM T64553 CS2I1H 5329217 IC50 = 6000 nM T64553 CQ70YG 5329218 IC50 = 5000 nM T64553 C6OL3X 5329220 IC50 = 4000 nM T64553 C2J4ZO 5329221 IC50 = 2000 nM T64553 CO87DJ 5329222 IC50 = 4000 nM T64553 C5LW1G 5329223 IC50 = 5000 nM T64553 CRB3S4 5329224 IC50 = 3000 nM T64553 CU68QR 5329225 IC50 = 2000 nM T64553 C4P7QH 5329226 IC50 = 3000 nM T64553 CWF7K8 5329227 IC50 = 2000 nM T64553 CJ6VE0 5329228 IC50 = 1000 nM T64553 C7WI1P 6326454 IC50 = 33000 nM T64553 CLB02J 6326455 IC50 = 14000 nM T64553 CZK47S 6326456 IC50 = 72000 nM T64553 CS23WK 6326457 IC50 = 7000 nM T64553 CR59JT 6326458 IC50 = 61000 nM T64553 CN1GO8 6326459 IC50 = 5000 nM T64553 CY4WT0 6326460 IC50 = 3000 nM T64553 CEW21T 6326461 IC50 = 6000 nM T64553 C3PNU9 6326462 IC50 = 6000 nM T64553 CLTQ35 6326463 IC50 = 5000 nM T64553 CU6S2L 6326464 IC50 = 6000 nM T64553 CP0XI6 6603792 IC50 > 50000 nM T64553 CTR6H5 9817349 IC50 = 5200 nM T64553 CXQ9J0 9856983 Ki = 419.1 nM T64553 C9JC1G 9866765 IC50 = 250 nM T64553 CM5Z8X 9869943 IC50 = 400 nM T64553 CR2B8U 9888491 IC50 = 54 nM T64553 CKZ8E3 9905577 IC50 = 7200 nM T64553 CG6A1H 9927800 IC50 = 1900 nM T64553 CKSC41 9939626 IC50 = 25000 nM T64553 C84LCW 9985193 IC50 = 22000 nM T64553 CSMY08 9988860 IC50 = 320 nM T64553 CUY0F8 10005715 IC50 = 47 nM T64553 CGOT13 10022152 IC50 = 8300 nM T64553 C4JO8F 10028975 IC50 = 41 nM T64553 C1O4GZ 10031003 IC50 = 7000 nM T64553 CUJR40 10062694 EC50 > 2000 nM T64553 CF1D6Y 10075240 IC50 = 88 nM T64553 CCW7U3 10097544 IC50 = 600 nM T64553 CM2VB6 10100735 IC50 > 500000 nM T64553 C97GRN 10248747 IC50 = 80000 nM T64553 CCQ2N6 10253089 IC50 = 230 nM T64553 C7SFI1 10296883 IC50 > 10000 nM T64553 CP4M1C 10347718 IC50 = 18000 nM T64553 C24LNX 10457649 IC50 = 160 nM T64553 CDQO71 10461517 IC50 > 500000 nM T64553 CNBX16 11270660 IC50 > 10000 nM T64553 CMXI90 11324412 Ki = 270 nM T64553 CJC95A 11454205 IC50 > 50000 nM T64553 CACS26 11561968 Ki > 2000 nM T64553 C5B3XJ 11620410 IC50 > 25000 nM T64553 C9ZD2E 11626406 IC50 = 3272 nM T64553 CJ9KN7 11683817 IC50 > 10000 nM T64553 CP3U0W 11684933 IC50 = 992 nM T64553 CU0E8O 11690457 Ki > 2000 nM T64553 CP7AH3 11755812 IC50 = 50000 nM T64553 CS36BH 11843159 IC50 = 370 nM T64553 C9JT4S 11847343 IC50 > 10000 nM T64553 CHR92S 11858109 IC50 > 8300 nM T64553 COS89C 12017518 IC50 = 6500 nM T64553 COIJ48 12968819 IC50 = 198000 nM T64553 C4AIU2 12968822 IC50 = 19000 nM T64553 CQ9Z0L 15550318 IC50 = 125 nM T64553 C5SDO8 15550319 IC50 = 424 nM T64553 CPZQ16 15550320 IC50 = 11 nM T64553 CK1ZB8 15550321 IC50 = 188 nM T64553 C9TU1O 16046126 IC50 > 1000 nM T64553 CKR57M 16086104 IC50 > 25000 nM T64553 C16NRY 16086114 IC50 > 25000 nM T64553 CQG45C 16109001 IC50 = 25000 nM T64553 C9MNP2 17549086 IC50 = 8600 nM T64553 CL9BQ6 17748275 IC50 = 25000 nM T64553 C3E1QT 18545586 IC50 = 4300 nM T64553 C7O1RC 18545605 IC50 = 26 nM T64553 C7TL8W 18545623 IC50 = 31 nM T64553 C06QRG 18545643 IC50 = 332 nM T64553 CX8GM1 18545657 IC50 = 46 nM T64553 CAN67W 20579088 IC50 = 396 nM T64553 C0E2OG 20579089 IC50 = 8 nM T64553 CJC5F3 20741385 Ki = 1551 nM T64553 CT39NL 22736235 IC50 > 50000 nM T64553 CA97TZ 22958832 IC50 = 13200 nM T64553 C7YG1N 24759534 IC50 > 100000 nM T64553 CAJ4T2 24762205 IC50 > 10000 nM T64553 C5ZM4T 24936119 IC50 > 10000 nM T64553 CS3Q8B 24995659 IC50 > 2000 nM T64553 CBK82P 25011729 IC50 > 30000 nM T64553 CQ67BO 25113172 Ki = 240 nM T64553 CK56UI 25138150 IC50 = 3000 nM T64553 CL0Q2A 25138151 IC50 = 10000 nM T64553 CHN12U 25138152 IC50 = 1900 nM T64553 CAU4D5 25138153 IC50 = 3500 nM T64553 CO6N7P 25138154 IC50 = 400 nM T64553 CT68EU 25138155 IC50 = 5500 nM T64553 C70QFH 25138156 IC50 = 5100 nM T64553 C12QZB 25138157 IC50 = 410 nM T64553 CL4I9B 25138158 IC50 = 930 nM T64553 C3J0NC 25138159 IC50 = 220 nM T64553 CTG9V4 25138160 IC50 = 530 nM T64553 CO59KB 25138161 IC50 = 340 nM T64553 C7EWQ6 25138162 IC50 = 910 nM T64553 CJ1IR3 25138163 IC50 = 150 nM T64553 CIL37K 25138164 IC50 = 920 nM T64553 CY2FZ5 25138165 IC50 = 200 nM T64553 C2JZV0 25138166 IC50 = 150 nM T64553 CB6H4P 25138167 IC50 = 190 nM T64553 C18JWR 25138168 IC50 = 420 nM T64553 CPJ61T 25138169 IC50 = 180 nM T64553 C2QSY5 25138170 IC50 = 660 nM T64553 CF12ZW 25138171 IC50 = 690 nM T64553 C5QR9L 25138172 IC50 = 3200 nM T64553 CQ5AR4 25138173 IC50 = 240 nM T64553 C08VAE 25138174 IC50 = 480 nM T64553 CID5O7 25169255 Ki = 318 nM T64553 CN2B0H 25169256 Ki = 677 nM T64553 CEL61X 44229839 IC50 > 10000 nM T64553 CJ3PF9 44313929 IC50 > 500000 nM T64553 CUV7K3 44313930 IC50 > 500000 nM T64553 CHK9N3 44313931 IC50 > 500000 nM T64553 CEKR19 44313990 IC50 > 500000 nM T64553 CD5PI9 44313997 IC50 = 441000 nM T64553 C5E4GK 44314373 IC50 > 500000 nM T64553 C3YD1G 44314380 IC50 > 500000 nM T64553 CPC68H 44314402 IC50 > 500000 nM T64553 C1RGE3 44315963 IC50 = 530000 nM T64553 CKN35W 44329183 IC50 = 1900 nM T64553 CM45BX 44329185 IC50 = 3200 nM T64553 CUN6G8 44329458 IC50 = 250 nM T64553 CX04DQ 44332978 IC50 = 40000 nM T64553 C1Z2NI 44353160 IC50 = 100000 nM T64553 CIG07A 44353173 IC50 > 100000 nM T64553 CB3K6R 44353260 IC50 = 100000 nM T64553 CY6PX0 44353421 IC50 = 100000 nM T64553 CX6A7T 44353525 IC50 > 100000 nM T64553 C3PGO1 44353601 IC50 = 63000 nM T64553 CZ2YC5 44353697 IC50 = 38 nM T64553 C8NBI3 44353815 IC50 = 422000 nM T64553 C8J1NC 44353827 IC50 > 500000 nM T64553 C8FVG3 44353828 IC50 = 328000 nM T64553 CG56OR 44565801 IC50 = 8400 nM T64553 C2XR9S 44578584 IC50 = 6400 nM T64553 CE98FP 44578585 IC50 = 9000 nM T64553 C4GJX8 44578586 IC50 = 1100 nM T64553 C15IVX 44578626 IC50 = 50000 nM T64553 C6RPJ3 44578627 IC50 = 26000 nM T64553 C39XME 44578661 IC50 = 110 nM T64553 C9TZE1 44578662 IC50 = 120 nM T64553 C0YMS8 44578663 IC50 = 97 nM T64553 CAYN97 44588971 IC50 = 12400 nM T64553 CEL6D9 44588972 IC50 = 1800 nM T64553 CNZ2H5 44589000 IC50 > 10000 nM T64553 CCYQ91 44589001 IC50 = 230 nM T64553 CV5GD1 44589002 IC50 = 120 nM T64553 C83KEG 44589022 IC50 = 330 nM T64553 CTZX27 44589023 IC50 > 10000 nM T64553 C34KTW 44589024 IC50 = 1700 nM T64553 C59BIS 44589025 IC50 = 4100 nM T64553 C4TUK3 44589050 IC50 = 730 nM T64553 CNA20V 44589051 IC50 = 480 nM T64553 CA5UF3 44589514 Ki = 1000 nM T64553 C3KLD1 44589515 Ki = 680 nM T64553 C7A0UX 44589516 Ki = 1140 nM T64553 CYK07V 44589517 Ki = 750 nM T64553 C89COX 44590149 Ki = 2145 nM T64553 C2BQ4M 44590150 Ki = 754 nM T64553 C6NB9K 44590204 Ki = 410 nM T64553 CQ0NU8 44590205 Ki = 450 nM T64553 C87MBD 44593467 IC50 = 3300 nM T64553 CZ20KC 44593469 Ki = 3500 nM T64553 CM3T7B 44593470 Ki = 560 nM T64553 CD2FE4 44593471 Ki = 1030 nM T64553 CS8GE3 44593472 Ki = 891 nM T64553 CKM4H0 44593475 Ki = 1500 nM T64553 CU3RF1 45139989 IC50 > 10000 nM T64553 CQGZ06 45139991 IC50 > 10000 nM T64553 CY83PR 45267327 IC50 > 1000 nM T64553 C84QFJ 45269074 IC50 = 200 nM T64553 C3DH8I 45273358 IC50 > 1000 nM T64553 CY8FI4 45482611 IC50 = 10 nM T64553 C8R0QT 45482612 IC50 = 90 nM T64553 C4QJY8 45482613 IC50 = 130 nM T64553 C23KBC 45482614 IC50 = 300 nM T64553 CGU1D9 45482615 IC50 = 400 nM T64553 CW0O3A 45482616 IC50 = 530 nM T64553 CJY07T 45482618 IC50 = 40 nM T64553 COTG54 45482619 IC50 = 170 nM T64553 CGZI81 45482621 IC50 = 50 nM T64553 C0Z2CA 45482622 IC50 = 70 nM T64553 CDA12W 45482623 IC50 = 700 nM T64553 CBFR47 45482624 IC50 = 80 nM T64553 CNW3O0 45482625 IC50 = 200 nM T64553 CO7EL4 45482626 IC50 = 1200 nM T64553 CV2F8C 45482627 IC50 = 1700 nM T64553 CX2J8I 45482628 IC50 = 2000 nM T64553 CAV67Y 45482629 IC50 = 3000 nM T64553 CI3B2P 45482637 IC50 = 50000 nM T64553 CPK9H0 45482644 IC50 = 10 nM T64553 C53KDV 45482647 IC50 = 280 nM T64553 C1GSJ3 45482648 IC50 = 1800 nM T64553 C37RUW 45482653 IC50 = 3000 nM T64553 CRL9P2 45482656 IC50 = 10000 nM T64553 CET79H 45493316 IC50 = 62000 nM T64553 C1J6GR 46224908 IC50 > 10000 nM T64553 C7ON5A 46233287 IC50 > 10000 nM T64553 CC2O9R 46865656 IC50 = 19952.62 nM T64553 C60GAV 46929544 IC50 > 8000 nM T64553 CP34VL 46929748 IC50 > 1000 nM T64553 CJ2E9Q 46929857 IC50 > 25000 nM T64553 CHSF07 49806372 IC50 > 1000 nM T64553 CF91RS 49843531 IC50 > 10000 nM T64553 C2Y6QS 50938552 IC50 > 10000 nM T64553 C9NYP4 51036677 IC50 > 10000 nM T64553 C4WRY3 51037112 IC50 > 10000 nM T64553 CRI28Z 51037948 IC50 > 10000 nM T64553 CEQN27 52936621 Ki > 2000 nM T64553 C2W9OA 53324451 IC50 > 10000 nM T64553 CD4H3S 53354074 Ki > 1000 nM T64553 C8NA4L 53384644 IC50 > 30000 nM T64553 CT3EW2 59292007 IC50 > 1000 nM T64553 CXJ63M 59603829 IC50 > 100000 nM T64553 CQEU96 59603842 IC50 > 10000 nM T64553 COH62U 60097413 IC50 > 3300 nM T64553 C1MR8Q 60097495 IC50 > 5000 nM T64553 CSZ6I5 66556035 IC50 = 100 nM T64553 CV63UL 67240318 IC50 > 10000 nM T64553 C8I7GC 68293638 IC50 > 10000 nM T64553 CD56XK 68293660 IC50 > 10000 nM T64553 C5DGR9 69036886 IC50 = 10000 nM T64553 CEBO91 71452977 IC50 > 10000 nM T64553 CI71DK 71533675 IC50 = 5.3 nM T64553 CCN01X 71547862 IC50 > 10000 nM T64553 CZ31PU 71583657 IC50 > 10000 nM T64553 CS62NH 71698376 IC50 = 53850 nM T64553 CI8X1R 71698379 IC50 = 995800 nM T64553 CKMZ39 72202597 IC50 = 251 nM T64553 CZ97VP 86294733 IC50 = 340 nM T64553 CS7GX8 89708625 IC50 = 73420 nM T64553 C1HW4B 89735655 IC50 > 100000 nM T64553 CY0UC4 90645194 IC50 > 10000 nM T64553 CV9H8U 90656285 IC50 = 18 nM T64553 CG7E1U 90656286 IC50 = 350 nM T64553 CDF9O2 90656287 IC50 = 81 nM T64553 CF89DA 90664659 IC50 = 11200 nM T64553 CCVL49 100942265 IC50 = 30000 nM T64553 CY7BI2 118706214 IC50 > 10000 nM T64553 C08KEM 122179540 IC50 = 6400 nM T64553 CG0RP7 122179547 IC50 = 5200 nM T64553 C1A0SQ 122179548 IC50 = 5500 nM T64553 CUO0C5 132156633 IC50 > 10000 nM T64553 CQS0J5 135494737 IC50 = 26000 nM T64553 C4SN0G 135548971 IC50 = 21000 nM T64553 CI47VJ 135566923 IC50 = 133 nM T64553 CHU3A2 135635724 IC50 = 8000 nM T64553 C29PWN 135886762 IC50 = 4000 nM T64553 CYDM01 135891431 IC50 > 1000 nM T64553 CHA4N2 136013680 IC50 > 10 nM T64553 CU9R3M 136036273 Ki = 1548.82 nM T64553 CHL5Z7 136056540 IC50 = 74 nM T64553 CO0L9T 136056541 IC50 = 33 nM T64553 CLIE18 136056542 IC50 = 815 nM T64553 CM7V8J 136056543 IC50 > 10000 nM T64553 C64BEV 136056544 IC50 = 14 nM T64553 CP1MX4 136056545 IC50 = 375 nM T64553 C4AR8N 136056546 IC50 = 445 nM T64553 CC10GD 136056547 IC50 = 3000 nM T64553 CN1PY3 136056548 IC50 = 47 nM T64553 CI8Y0U 136056549 IC50 > 10000 nM T64553 C1YUD0 136219394 IC50 > 10 nM T64553 CIU8W3 136254389 IC50 > 10 nM T64553 CLJH31 139209093 EC50 > 20000 nM T64553 CVI30A 139600340 EC50 = 41 nM T64553 C8TL1A 155513050 EC50 = 420 nM T64553 C2MD1Q 155513187 IC50 > 10000 nM T64553 CEDI24 155516854 EC50 = 49 nM T64553 CGDJ81 155539793 EC50 = 1400 nM T64553 CDW9G6 155541623 EC50 = 4050 nM T64553 CLJ80U 155548662 EC50 = 56 nM T64553 CGTR28 155552797 EC50 = 88 nM T64553 CCV06Q 155554126 EC50 = 42 nM T64553 C3DQI8 155557074 EC50 = 5700 nM T64553 CVS68Y 155558083 EC50 = 7900 nM T64553 CT8VX1 155562023 EC50 = 28 nM T64553 CR6EL3 155568078 EC50 = 2700 nM T64553 C12HQW 155568509 EC50 = 2000 nM T64553 D00SEC 3641059 Ki = 2630.27 nM T64553 D03DZO 11715767 IC50 > 10000 nM T64553 D03OKV 9844320 IC50 > 1000 nM T64553 D04PEI 11467730 IC50 > 50000 nM T64553 D06HVH 54613583 IC50 > 10000 nM T64553 D06WGX 9549184 IC50 > 25000 nM T64553 D07ADX 54764565 IC50 = 5050 nM T64553 D07OXC 11650194 IC50 > 5400 nM T64553 D08HFG 24809764 IC50 > 10000 nM T64553 D09HVH 135566652 IC50 > 10 nM T64553 D0A0JL 2052 Ki > 10000 nM T64553 D0E1QI 9549297 Ki > 10000 nM T64553 D0J3LR 11634725 Ki > 4000 nM T64553 D0OZ2S 11785878 IC50 = 1500 nM T64553 D0P6JS 11675054 IC50 > 10000 nM T64553 D0R2WK 16038120 IC50 = 1598 nM T64553 D0T4MJ 9549296 IC50 = 11200 nM T64553 D0Y5RO 4566 Ki > 10000 nM T42247 D07CLV 46940575 Ki < 50 nM T42247 CFXK28 11497354 Ki = 40000 nM T42247 CQY48M 44820626 Ki = 110000 nM T42247 C0E9LP 44820627 Ki = 53000 nM T42247 C3XU7D 46830176 Ki = 130000 nM T42247 CL75NA 46883825 Ki = 160000 nM T42247 C2QPO5 46883826 Ki = 160000 nM T42247 CXT0Z7 46883827 Ki = 140000 nM T42247 CL3QR5 46883828 Ki = 140000 nM T42247 C6HNB8 46883881 Ki = 2700000 nM T42247 CF2O4P 46883882 Ki = 2800000 nM T42247 C6O1UC 46883883 Ki = 710000 nM T42247 C7JAQ0 46883921 Ki = 200000 nM T42247 CKUQ91 46883922 Ki = 460000 nM T42247 CW1PR3 46883923 Ki = 730000 nM T42247 C3SZP1 46883924 Ki = 140000 nM T42247 C8Z2MB 46883992 Ki = 68000 nM T42247 C8RBO6 46883993 Ki = 130000 nM T42247 CH92NU 46883994 Ki = 130000 nM T42247 CN0P3Q 46884021 Ki = 44000 nM T42247 C1DS6K 46884022 Ki = 36000 nM T42247 C90AVJ 46884023 Ki = 49000 nM T42247 C49JKQ 46884084 Ki = 32000 nM T42247 CPB9H7 46884085 Ki = 24000 nM T42247 CD7AG0 46884409 Ki = 1200000 nM T42247 CF3QO9 46884410 Ki = 220000 nM T42247 CLZ07E 46884435 Ki = 100000 nM T42247 C2GB8Y 46884436 Ki = 68000 nM T42247 C40MQS 46884474 Ki = 45000 nM T42247 C8Q0RI 46884475 Ki = 180000 nM T42247 CE62KI 46884476 Ki = 200000 nM T42247 C0E5CW 46884477 Ki = 130000 nM T42247 C8RL0W 46884520 Ki = 120000 nM T42247 CM1D9E 46884521 Ki = 68000 nM T42247 C9X6JF 46884522 Ki = 210000 nM T42247 C59USH 46884523 Ki = 69000 nM T97873 D0K3UQ 10343454 Ki = 1.1 nM T97873 C5DU0L 1448028 IC50 = 232 nM T97873 C1USE0 58398295 IC50 > 10000 nM T97873 C5KT7M 91810833 Ki = 3 nM T97873 C6ENV5 100951623 IC50 > 10000 nM T97873 CJ8P9N 118197423 Ki = 13 nM T97873 CX56WS 118197424 Ki = 189 nM T97873 C9G7DJ 118197428 Ki = 6 nM T97873 C2C3FW 118197452 Ki = 3 nM T97873 CM0OR7 118197461 Ki = 78 nM T97873 CY9VS3 118197480 Ki = 22 nM T97873 CV96SI 118197481 Ki = 16 nM T97873 C35CDF 118197490 Ki = 25 nM T97873 CFC3U5 118197510 Ki = 30 nM T97873 CL45BZ 118197515 Ki = 19 nM T97873 CWU50A 118197518 Ki = 618 nM T97873 CX1O5U 118197542 Ki = 22 nM T97873 CKJ51V 118197543 Ki = 100 nM T97873 CB2MR1 118197598 Ki = 479 nM T97873 CVB8G2 118204555 Ki = 13 nM T97873 C1DI4U 118204557 Ki = 14 nM T97873 CRIG68 118204583 Ki = 2713 nM T97873 CQN31U 118204585 Ki = 123 nM T97873 C2QSG1 118204586 Ki = 1322 nM T97873 C16WRU 118204596 Ki = 54 nM T97873 C0J9SL 118204597 Ki = 31 nM T97873 C4I3MX 118204598 Ki = 45 nM T97873 CI2O9F 118204599 Ki = 8 nM T97873 CD8FK4 118204600 Ki = 30 nM T97873 CC9QH3 118204611 Ki = 7 nM T97873 C19JMW 118204615 Ki = 24 nM T97873 C9Q2RN 118204621 Ki = 6 nM T97873 CKHO92 118204622 Ki = 5 nM T97873 CFU29O 118204628 Ki = 23 nM T97873 C3HKS9 118204630 Ki = 2 nM T97873 C64JPL 118204633 Ki = 7 nM T97873 C14RPE 118204645 Ki = 128 nM T97873 CM2L1Y 118204648 Ki = 16 nM T97873 CP1QM2 118204670 Ki = 16 nM T97873 CHPL62 118204671 Ki = 9 nM T97873 CI4MB6 118204681 Ki = 51 nM T97873 C4WAU6 118204692 Ki = 20 nM T97873 CKJ13S 118204706 Ki = 28 nM T97873 C6XZ4L 118204712 Ki = 85 nM T97873 C5CLA7 118204739 Ki = 78 nM T97873 CKZ49G 118204744 Ki = 22 nM T97873 CN7A2B 118204755 Ki = 206 nM T97873 CO4U7S 118204758 Ki = 21 nM T97873 CALE90 118204759 Ki = 8 nM T97873 CME93A 118204768 Ki = 19 nM T97873 C4TQ9B 118204773 Ki = 108 nM T97873 CO6TZ5 118204799 Ki = 10 nM T97873 CU26QH 118204818 Ki = 11 nM T97873 CQ95YK 118204826 Ki = 58 nM T97873 C8OWM0 118204829 Ki = 5 nM T97873 CY1F7E 118204847 Ki = 456 nM T97873 C9CR2G 118204853 Ki = 19 nM T97873 CEZ7Y3 118204870 Ki = 25 nM T97873 C4JFT8 118204879 Ki = 22 nM T97873 C0GU3M 118204881 Ki = 11 nM T97873 C1DJ4F 118204898 Ki = 59 nM T97873 C60QYJ 118204900 Ki = 6 nM T97873 C9B8QU 118204904 Ki = 123 nM T97873 CU7DY1 118204918 Ki = 73 nM T97873 CHY89U 118205008 Ki = 18 nM T97873 CA2V4B 122185738 IC50 = 2500 nM T97873 C0FSC3 122185739 IC50 = 958 nM T97873 C5T8CN 122185740 IC50 = 29 nM T97873 CP58TW 122185741 IC50 = 95 nM T97873 C3N2MR 122185742 IC50 = 89 nM T97873 CIA68E 122185743 IC50 = 3163 nM T97873 C4ZQ3S 122185744 IC50 = 3477 nM T97873 C4ZPQ2 122185745 IC50 = 491 nM T97873 CIK57S 122185746 IC50 = 52 nM T97873 C0QLZ2 122185747 IC50 = 8.7 nM T97873 C8WVG7 122185748 IC50 = 0.3 nM T97873 CR2E1O 122185749 IC50 = 3.2 nM T97873 CH2G4O 122185750 IC50 = 3.2 nM T97873 CQ8IU6 122185751 IC50 = 3.8 nM T97873 CRK1C7 122185752 IC50 = 11 nM T97873 CY4KC3 122185753 IC50 = 4 nM T97873 C7NV8I 122185754 IC50 = 27 nM T97873 CM01KN 122185755 IC50 = 214 nM T97873 CLX65V 122185756 IC50 = 14 nM T97873 CN1H7Z 122185757 IC50 = 9 nM T97873 CM10NT 122185758 IC50 = 26 nM T97873 CBPE58 122185759 IC50 = 11 nM T97873 CBY08V 122185760 IC50 = 6 nM T97873 CMS57L 122185761 IC50 = 25 nM T97873 CJ4K3S 122185762 IC50 = 421 nM T97873 COB25C 122185763 IC50 = 170 nM T97873 C40GPQ 122185764 IC50 = 614 nM T97873 C94IYK 122185765 IC50 = 3604 nM T97873 C4KP5E 122185766 IC50 = 812 nM T97873 C9W2NU 122185767 IC50 = 268 nM T97873 CMVF34 122185768 IC50 = 1005 nM T97873 CA2XJ8 122185769 IC50 = 715 nM T97873 CJDN65 123327510 Ki = 30 nM T97873 CYJ3D6 123416489 Ki = 12 nM T97873 C0FAL9 123776529 Ki = 18 nM T97873 CS6R2Y 123866952 Ki = 13 nM T97873 CO2C1L 124167959 Ki = 6 nM T97873 C1Q8XU 124167985 Ki = 4 nM T97873 CL03NI 127048631 IC50 = 36 nM T97873 C4VG5S 127049670 IC50 = 8 nM T97873 C9W1BL 127049671 IC50 = 8400 nM T97873 C5BJX0 127049672 IC50 = 29 nM T97873 C9GSP5 127049673 IC50 = 93 nM T97873 C9ZT2F 127049674 IC50 = 451 nM T97873 C2R7MO 127049675 IC50 = 277 nM T97873 C13MYW 127049676 IC50 = 1.5 nM T97873 C25YWZ 127049978 IC50 = 50000 nM T97873 C9S5ZK 127050864 IC50 = 232 nM T97873 CHL64W 127051187 IC50 > 10000 nM T97873 C7B8QY 127051188 IC50 = 85 nM T97873 C08CTU 127051189 IC50 = 75 nM T97873 CS6X7K 127053022 IC50 = 378 nM T97873 C0YAN3 127053023 IC50 = 111 nM T97873 CZ2MK8 127053024 IC50 = 207 nM T97873 CZ69TS 127053025 IC50 = 35 nM T97873 CGW81F 127053026 IC50 = 113 nM T97873 CUG2X5 127053027 IC50 = 70 nM T97873 D06MBD 11176403 IC50 < 3000 nM T65818 CDBF98 281242 Ki = 16900 nM T65818 C6L1VE 1551321 Ki > 250000 nM T65818 C4BKQ3 4798291 IC50 > 200000 nM T65818 CUX8S7 7197248 IC50 < 1000000 nM T65818 CN5H0B 10970861 Ki = 1040 nM T65818 C5OPG0 11127644 Ki > 250000 nM T65818 C10KPB 11142955 Ki = 350 nM T65818 CF19DX 13509139 Ki = 106000 nM T65818 C4Y1HP 15849848 Ki > 250000 nM T65818 CVRO49 25760265 IC50 = 81200 nM T65818 CX18KT 44447089 Ki = 1030 nM T65818 CO34LD 45464518 IC50 = 140000 nM T65818 CN53IO 53792079 Ki = 8190 nM T65818 CT9PG8 71457393 IC50 > 100000 nM T65818 C7P2UD 71817806 IC50 = 11500 nM T65818 CMQN63 71817809 IC50 = 24900 nM T65818 C1N7QD 71817963 IC50 > 100000 nM T65818 CMBJ36 71817964 IC50 = 23900 nM T65818 CK2T9X 71817965 IC50 > 100000 nM T65818 CE7VJ4 71817966 IC50 > 100000 nM T65818 C74CNV 72193911 IC50 = 11 nM T65818 CU8WB9 73437637 IC50 = 159000 nM T65818 CRU02V 74766022 Ki = 47000 nM T65818 CJ2UC1 85470733 IC50 > 200000 nM T65818 CRA08X 85470742 IC50 > 200000 nM T65818 C05HWU 86140993 Ki > 250000 nM T65818 CR0PF5 86222557 IC50 = 160000 nM T65818 CF35LZ 87495845 Ki > 250000 nM T65818 C81VCX 110482493 IC50 > 100000 nM T65818 CVS60Z 118720629 Ki = 7670 nM T65818 C4VWL9 118720630 Ki = 152 nM T65818 C71CKB 118720631 Ki = 4570 nM T65818 CCQ74S 118720632 Ki = 2180 nM T65818 C8JDP5 118720633 Ki = 185 nM T65818 CE9X4G 118720634 Ki = 205 nM T65818 CW87DK 118720635 Ki = 241 nM T65818 CKIF61 118720636 Ki > 250000 nM T65818 CJ6MY3 118720637 Ki > 250000 nM T65818 CP5V7M 118720638 Ki > 250000 nM T65818 CU5F3O 118734160 IC50 > 100000 nM T65818 CB67XZ 118734161 IC50 = 3200 nM T65818 C5HV4G 118734165 IC50 = 9800 nM T65818 CB7W1N 118734166 IC50 = 3700 nM T65818 CVQ9B5 118734167 IC50 > 100000 nM T65818 C3VMB4 118734170 IC50 = 2600 nM T65818 C5B3AO 118734171 IC50 = 4500 nM T65818 CR02XN 118734172 IC50 = 4800 nM T65818 CYQ61P 118734173 IC50 = 13000 nM T65818 CD6IM0 118734175 IC50 = 52000 nM T65818 CG1NJ3 118734176 IC50 = 2100 nM T65818 CTL4C9 118734177 IC50 = 8300 nM T65818 C1UWG8 118734178 IC50 = 17000 nM T65818 CWK18R 118734179 IC50 = 50000 nM T65818 CED26H 118734180 IC50 > 100000 nM T65818 C24VOF 118734181 IC50 = 33000 nM T65818 C3KJR9 118734182 IC50 = 39000 nM T65818 CMWH70 118734252 IC50 = 40000 nM T65818 CS1R6T 118734253 IC50 > 100000 nM T65818 CK3NV4 118734254 IC50 > 100000 nM T65818 C4VK6O 118734255 IC50 > 100000 nM T65818 C7AH4D 118734256 IC50 > 100000 nM T65818 CZ04FM 118734257 IC50 > 100000 nM T65818 CZ97HL 118734258 IC50 = 6400 nM T65818 C1DKP8 118734259 IC50 = 1600 nM T65818 CET0D8 118734260 IC50 = 3800 nM T65818 C4N7KF 118734261 IC50 = 2500 nM T65818 C2M4UZ 118734262 IC50 = 5000 nM T65818 C3PL1T 118734263 IC50 = 518 nM T65818 C3OS1H 118734264 IC50 = 589 nM T65818 C9NWC0 118734265 IC50 = 58000 nM T65818 CX0OA9 118734267 IC50 = 58000 nM T65818 CU8I4F 118734268 IC50 = 1100 nM T65818 CI6S8L 118734269 IC50 = 2500 nM T65818 CH2LO8 118734272 IC50 > 100000 nM T65818 CI9RT3 118734273 IC50 = 1900 nM T65818 C3KLH4 118734276 IC50 > 100000 nM T65818 CPUI84 118734277 IC50 > 100000 nM T65818 C96PKA 118734278 IC50 = 5500 nM T65818 C4AL9Z 118734279 IC50 = 11000 nM T65818 C71TGN 118734280 IC50 = 11800 nM T65818 C8V9EB 118734281 IC50 = 16000 nM T65818 CIZ3Q6 118734282 IC50 = 15100 nM T65818 CJ64ZC 118734283 IC50 = 20500 nM T65818 C1K7AN 118734284 IC50 = 4800 nM T65818 C6XY9M 118734285 IC50 > 100000 nM T65818 CY8X0V 118734286 IC50 = 70000 nM T65818 CO4F3Y 118734287 IC50 = 9400 nM T65818 C9CN6S 118734288 IC50 = 21000 nM T65818 CN7SR4 118734290 IC50 = 6200 nM T65818 C57ZSG 118734291 IC50 = 38000 nM T65818 CKST54 118734292 IC50 = 755 nM T65818 C9XDY5 118734293 IC50 = 709 nM T65818 C01PYL 118734294 IC50 = 237 nM T65818 CO6PR7 118734295 IC50 = 30600 nM T65818 C4ZPC8 118734296 IC50 = 1400 nM T65818 CJ40TN 118734297 IC50 = 1100 nM T65818 CA9X0N 118734298 IC50 = 11800 nM T65818 C7FMV5 126456392 Ki = 200 nM T65818 C7UJ4W 127043855 IC50 = 550 nM T65818 CW0FZ2 127044995 Ki = 65200 nM T65818 C06JOP 127044996 Ki > 250000 nM T65818 CM0VT4 127048200 Ki > 250000 nM T65818 CTL4Z8 127048201 Ki = 55300 nM T65818 CBQ4S3 127048202 Ki = 7940 nM T65818 CC96VU 127048834 Ki > 250000 nM T65818 CTY5D4 127049157 Ki = 622 nM T65818 CF3HO2 127049196 Ki = 10300 nM T65818 C03XKF 127049491 Ki > 250000 nM T65818 CFW6M1 127049492 Ki > 250000 nM T65818 CL6D0Z 127049497 Ki = 3020 nM T65818 C4I1RH 127049824 Ki = 10600 nM T65818 C2A1MZ 127050130 Ki = 1020 nM T65818 CA4MP3 127050430 Ki = 5540 nM T65818 CJT5R9 127050433 Ki = 7700 nM T65818 C0N2LE 127050745 Ki = 11500 nM T65818 C9GBD2 127051304 Ki = 24900 nM T65818 CLK50R 127051701 Ki = 9510 nM T65818 C2BUZ7 127051959 Ki = 8230 nM T65818 CK81ME 127051999 Ki = 1300 nM T65818 CAC25R 127052273 Ki = 632 nM T65818 C3FMN7 127052612 Ki = 3470 nM T65818 CHA9Q6 127052870 Ki = 1680 nM T65818 CJM96B 127053163 Ki = 1420 nM T65818 C8QO7V 135554374 IC50 = 34000 nM T65818 CXLS30 137633011 IC50 = 128 nM T65818 CMC5E8 137634250 IC50 = 190 nM T65818 CER06G 137637900 IC50 = 13814 nM T65818 C97XKO 137638141 IC50 = 246 nM T65818 CMTG53 137639983 IC50 = 129 nM T65818 CH6DQ2 137640549 IC50 = 4622 nM T65818 C9SWV7 137640590 IC50 = 412 nM T65818 CG0ED2 137641900 IC50 = 144 nM T65818 C3SP9K 137642894 IC50 = 2565 nM T65818 C1U3ZM 137642974 IC50 = 271 nM T65818 CYN9Z5 137646376 IC50 = 225 nM T65818 CDU93R 137646849 IC50 = 130 nM T65818 C96EWT 137647165 IC50 = 118 nM T65818 CJM57W 137648545 IC50 = 123 nM T65818 CC9T7O 137650040 IC50 = 83 nM T65818 CN9F2A 137650752 IC50 = 211 nM T65818 CB9VI7 137652734 IC50 = 96 nM T65818 CSM3V5 137653412 IC50 = 1922 nM T65818 CVI87E 137654495 IC50 = 105 nM T65818 C8DV5C 137655020 IC50 = 243 nM T65818 C2RIG6 137655030 IC50 = 56 nM T65818 CMT56C 137655972 IC50 = 878 nM T65818 C13POW 137656080 IC50 = 2271 nM T65818 CCTK37 137657323 IC50 = 345 nM T65818 C4VS2D 137658289 IC50 = 217 nM T65818 CKHE71 137659752 IC50 = 84 nM T65818 C0ID7T 137660529 IC50 = 37 nM T65818 C8E6UD 137661774 IC50 = 55 nM T65818 CV2U0Z 137662110 IC50 = 109 nM T65818 CJ47OK 145925583 Ki = 17700 nM T65818 CB1J0U 145994843 Ki = 27400 nM T65818 C94BDA 155510769 IC50 > 200000 nM T65818 CJMO47 155512116 Ki = 4900 nM T65818 CYE4R8 155512732 IC50 > 200000 nM T65818 CK9D4I 155512960 IC50 > 200000 nM T65818 C0CYS7 155515712 IC50 > 200000 nM T65818 C7VYT6 155517480 IC50 > 200000 nM T65818 CIH73R 155523459 IC50 > 10000 nM T65818 CD0F5Z 155524591 IC50 <= 200000 nM T65818 CGOU03 155531602 IC50 > 10000 nM T65818 CY1MF9 155534671 IC50 > 200000 nM T65818 C8E6QH 155538090 Ki = 17400 nM T65818 CZG6O5 155539882 IC50 > 200000 nM T65818 C8XYO7 155545269 Ki = 1200 nM T65818 C8R0JW 155547335 IC50 > 158489.32 nM T65818 CXP60U 155547553 Ki = 21400 nM T65818 CF35ER 155548478 IC50 = 740 nM T65818 CQM59I 155550629 Ki = 4300 nM T65818 COR09W 155554600 Ki = 700 nM T65818 CRU97I 155558560 IC50 > 10000 nM T65818 CRVJ23 155564248 Ki = 4800 nM T65818 CU0W9L 155566815 IC50 > 200000 nM T65818 CHEX85 445715 Ki > 250000 nM T65818 D02MNM 71817810 IC50 = 8900 nM T10822 D0W5HK 216239 IC50 = 199 nM T10822 D0M9QZ 11485656 IC50 = 14 nM T10822 C5E3BR 3835861 IC50 = 500 nM T10822 CN08CJ 11561907 IC50 = 12 nM T10822 C5VPH9 16129448 IC50 > 10000 nM T10822 C4KVF9 21039588 EC50 = 200 nM T10822 CCL3R5 49867929 IC50 = 4200 nM T10822 CD3G9X 59088919 EC50 = 25 nM T10822 C37NKO 67129970 IC50 = 2110 nM T10822 CK80LJ 67130050 IC50 > 10000 nM T10822 C7GRV2 68755406 IC50 > 10000 nM T10822 CRY5G3 70030697 EC50 = 1300 nM T10822 C1OW2Y 70031419 EC50 > 10000 nM T10822 C4VW9G 72548521 IC50 = 2450 nM T10822 CR18AC 72548523 IC50 = 415 nM T10822 CLJ7G8 72548748 IC50 = 1650 nM T10822 CX7OZ0 72705882 IC50 = 100 nM T10822 CQ2MF5 72705885 IC50 = 290 nM T10822 C10QBN 73776232 IC50 = 4.4 nM T10822 CBV89M 74221936 IC50 = 2.1 nM T10822 CP97AI 74221937 IC50 = 2.8 nM T10822 C3ST0F 74222016 IC50 = 1.9 nM T10822 C5W7FG 74222104 IC50 = 9.5 nM T10822 CTR9P7 74222108 IC50 = 11.4 nM T10822 CX9L1A 74222191 IC50 = 5 nM T10822 C74SUP 74222276 IC50 = 2.3 nM T10822 CZV0D1 74222277 IC50 = 2.3 nM T10822 CO3B2P 74222520 IC50 = 12.1 nM T10822 C85NSA 74222522 IC50 = 9.3 nM T10822 C2A1YD 74222612 IC50 = 5.5 nM T10822 CT8Z9V 74222614 IC50 = 3.3 nM T10822 C7QD4Z 74222786 IC50 = 16.4 nM T10822 CJC5U3 74222788 IC50 = 29.5 nM T10822 CRE2U3 77050682 IC50 = 7.2 nM T10822 C5KMS7 90340155 IC50 = 15 nM T10822 C9HFU5 91827689 IC50 = 0.6 nM T10822 C8W9KV 91844733 IC50 = 1200 nM T10822 CX3OS0 117072459 IC50 = 1.7 nM T10822 CXM12Z 117072461 IC50 = 2.3 nM T10822 CND7I4 117072462 IC50 = 49.2 nM T10822 CI6CU8 117995570 IC50 > 10000 nM T10822 CZAG19 117995615 IC50 > 10000 nM T10822 CO6I0P 118002788 IC50 = 4200 nM T10822 C7GWF6 118002790 IC50 = 4000 nM T10822 CJN7O1 118394955 IC50 = 17.5 nM T10822 CR5MY6 118394959 IC50 = 12 nM T10822 C87KJZ 118394996 IC50 = 2.7 nM T10822 CW1XY4 118395000 IC50 = 4.2 nM T10822 CEFB09 118395090 IC50 = 3.9 nM T10822 CZFR25 118395096 IC50 = 5.5 nM T10822 C4JO1G 118395100 IC50 = 32.8 nM T10822 C2OR0U 118395125 IC50 = 7 nM T10822 CW2HS7 118395147 IC50 = 20.5 nM T10822 C3N5HL 118407984 IC50 = 4.5 nM T10822 C43GUJ 118407987 IC50 = 14.7 nM T10822 C0A1PW 118408035 IC50 = 1.6 nM T10822 CXD69P 118408040 IC50 = 20.6 nM T10822 C8Y5KV 118408043 IC50 = 4.3 nM T10822 C1BU8L 118408129 IC50 = 3.2 nM T10822 C2AEN3 118408131 IC50 = 2.4 nM T10822 CGDW02 118408137 IC50 = 3.8 nM T10822 C2PS0G 118408140 IC50 = 2.8 nM T10822 CK1Q2L 118660560 IC50 = 30 nM T10822 CNS83A 118660576 IC50 = 23.1 nM T10822 C1XM9Q 118660581 IC50 = 24 nM T10822 CWM17K 118660591 IC50 = 21 nM T10822 CJPY20 118660604 IC50 = 4.7 nM T10822 CINY29 118660605 IC50 = 17.9 nM T10822 CC8N3S 118660612 IC50 = 1.1 nM T10822 C0E9JN 118660621 IC50 = 1946 nM T10822 C8S7IZ 118660623 IC50 = 87 nM T10822 C9EO4F 118660637 IC50 = 70 nM T10822 CZ67PS 118660644 IC50 = 0.2 nM T10822 CH3X6A 118660651 IC50 = 9 nM T10822 CGUH83 118660670 IC50 = 16 nM T10822 CMQF56 118660673 IC50 = 4.6 nM T10822 CUPD10 118660675 IC50 = 43 nM T10822 CT0K5W 118660681 IC50 = 5.8 nM T10822 C94WCU 118660701 IC50 = 10.7 nM T10822 CI75VN 118660710 IC50 = 559 nM T10822 CF5NW1 118660717 IC50 = 12.6 nM T10822 CX0PZ6 118660721 IC50 = 76 nM T10822 CQ68OU 118660724 IC50 = 19.4 nM T10822 CRJ1U0 118660735 IC50 = 590 nM T10822 C8DST2 118660737 IC50 = 11.2 nM T10822 C3H1EQ 118660753 IC50 = 87 nM T10822 CMHN53 118660754 IC50 = 45 nM T10822 C8L0EH 118660757 IC50 = 1418 nM T10822 C04SZP 118660758 IC50 = 34 nM T10822 CQIG81 118660764 IC50 = 16 nM T10822 CW1NF7 118660774 IC50 = 7.3 nM T10822 C5DS2P 118660778 IC50 = 2 nM T10822 CZ08CI 118660787 IC50 = 0.9 nM T10822 C6KPX5 118660788 IC50 = 73 nM T10822 C3AOC4 118660806 IC50 = 4.2 nM T10822 CC38NP 118660811 IC50 = 3.4 nM T10822 C10KTV 118660815 IC50 = 17.5 nM T10822 CR7UO0 118660828 IC50 = 396 nM T10822 C4C3OZ 118660833 IC50 = 9.9 nM T10822 C7RY4E 118660837 IC50 = 2.5 nM T10822 C26UWT 118660844 IC50 = 20.2 nM T10822 CVY97J 118660845 IC50 = 0.5 nM T10822 C5RWS7 118660850 IC50 = 27.8 nM T10822 CCZT29 118660866 IC50 = 8.2 nM T10822 C1GD2X 118660867 IC50 = 7.2 nM T10822 CVDE92 118660879 IC50 = 65 nM T10822 C7RI6Q 118660891 IC50 = 9.8 nM T10822 CD41TQ 118660893 IC50 = 4.7 nM T10822 CWD87S 118660909 IC50 = 0.6 nM T10822 CPD9X5 118660910 IC50 = 35.5 nM T10822 CI1F6B 118879399 IC50 = 230 nM T10822 C3C0ON 118879403 IC50 = 125 nM T10822 CI5QS0 118879418 IC50 = 120 nM T10822 CATC53 118879424 IC50 = 12 nM T10822 CWS41B 118879437 IC50 = 2.8 nM T10822 C4ZSV3 118879442 IC50 = 115 nM T10822 C8I6LD 118879477 IC50 = 19 nM T10822 CR0L5G 118879484 IC50 = 435 nM T10822 CCL26Y 118879516 IC50 = 800 nM T10822 CQ1TL7 118879520 IC50 = 28 nM T10822 CK7D6O 118879529 IC50 = 6.5 nM T10822 C9HZA6 118959784 IC50 = 25 nM T10822 CQG1Z6 118959791 IC50 = 76 nM T10822 CFM40Z 118959844 IC50 = 270 nM T10822 CIJ83N 118959880 IC50 > 10000 nM T10822 CO1S8J 118959907 IC50 = 82 nM T10822 C5XIA4 118959923 IC50 > 10000 nM T10822 CP3S7C 118959947 IC50 = 1900 nM T10822 C0FW6R 118959991 IC50 = 1500 nM T10822 CD8OQ1 118959995 IC50 = 710 nM T10822 CF2RI9 118960044 IC50 = 42 nM T10822 C03DZJ 118960049 IC50 = 53 nM T10822 CBRU31 118960075 IC50 = 140 nM T10822 CP21OJ 118960086 IC50 = 43 nM T10822 CX90DQ 118960168 IC50 = 94 nM T10822 C3LB2S 118960186 IC50 = 55 nM T10822 C03DNI 118960206 IC50 = 2000 nM T10822 CL8B9S 118960211 IC50 = 5 nM T10822 CHJ70O 118960212 IC50 = 49 nM T10822 C6AD9X 118960213 IC50 = 9 nM T10822 CWDN97 118960250 IC50 = 100 nM T10822 CM05PQ 118960252 IC50 = 13 nM T10822 CG2LU6 118960270 IC50 = 110 nM T10822 CFYW63 118960320 IC50 = 160 nM T10822 C1WQF4 118960328 IC50 = 27 nM T10822 CBCH81 118960335 IC50 = 313 nM T10822 C0WFS7 118974284 IC50 = 1900 nM T10822 CVW4H2 125487466 EC50 > 10000 nM T10822 CRM6E2 125487493 EC50 = 110 nM T10822 C6PHJ4 125501420 EC50 > 10000 nM T10822 CKXL61 125501579 EC50 = 9.1 nM T10822 CXJZ21 125501590 EC50 = 3 nM T10822 CO57LX 125501624 EC50 = 8.9 nM T10822 CEN34J 125501625 EC50 = 220 nM T10822 CI6Y7N 125501655 EC50 = 490 nM T10822 C9JIS1 125501676 EC50 = 66 nM T10822 C8XP9M 125501693 EC50 = 550 nM T10822 C8VOF9 125501698 EC50 = 0.77 nM T10822 CR8FA3 126511850 EC50 = 2.3 nM T10822 CSFJ98 126511854 EC50 = 1.3 nM T10822 CJ8ZB0 126511857 EC50 = 70 nM T10822 CL59RS 126511881 EC50 = 7.4 nM T10822 C8XE9S 126511887 EC50 = 2 nM T10822 CK07QF 126511899 EC50 = 2.6 nM T10822 CR1P4J 126511903 EC50 = 8.3 nM T10822 CNU6Y7 126511904 EC50 = 0.35 nM T10822 C25UMK 126511912 EC50 = 16 nM T10822 CN48PT 126511919 EC50 = 890 nM T10822 C20TLZ 126511932 EC50 = 3 nM T10822 CCY7X1 126511934 EC50 = 140 nM T10822 CL9T2O 126511947 EC50 = 0.58 nM T10822 CDPR40 126511985 EC50 = 1.5 nM T10822 CP4FI1 126511997 EC50 = 620 nM T10822 CR84ZE 126511999 EC50 = 0.4 nM T10822 CR29DV 126512018 EC50 = 1700 nM T10822 CN74DB 126512048 EC50 = 28 nM T10822 CP8DX9 126512116 EC50 > 10000 nM T10822 C7UQ5Y 126512118 EC50 = 1.4 nM T10822 C16LMU 126512125 EC50 = 2800 nM T10822 C28RUE 126512274 EC50 = 1400 nM T10822 CI0GZ9 126549930 EC50 = 21 nM T10822 C0NW9I 126568381 EC50 = 1300 nM T10822 C8E6SV 126568395 EC50 = 8.4 nM T10822 CAT7N0 126568404 EC50 = 84 nM T10822 C5JCA2 126568413 EC50 = 8.4 nM T10822 CD5Z4M 126568428 EC50 = 19 nM T10822 CL5K9W 126568459 EC50 = 11 nM T10822 CB0IM6 126568463 EC50 = 11 nM T10822 C2TV9X 126568478 EC50 = 110 nM T10822 CTH7Q8 126568496 EC50 = 21 nM T10822 C7GW6R 126568503 EC50 > 10000 nM T10822 CA3Z1S 126568509 EC50 = 14 nM T10822 CMTB82 126568548 EC50 = 2.3 nM T10822 CT49KO 126568570 EC50 = 12 nM T10822 CWH04B 126568590 EC50 = 28 nM T10822 C37ZWO 126568629 EC50 = 10 nM T10822 CXS70O 126568659 EC50 = 95 nM T10822 CEIX89 126568661 EC50 = 13 nM T10822 CJZB82 126568663 EC50 = 2.4 nM T10822 C8UXW1 126568668 EC50 = 3.1 nM T10822 C57AZT 126568669 EC50 = 16 nM T10822 CHRM10 126568696 EC50 = 690 nM T10822 CJD47X 126568714 EC50 = 140 nM T10822 CLZ1H3 126568746 EC50 = 27 nM T10822 CH8NT1 126568757 EC50 = 17 nM T10822 C0VES9 126568827 EC50 = 17 nM T10822 CAFZ61 126568853 EC50 = 150 nM T10822 C7DG0C 126568856 EC50 = 3.6 nM T10822 C0AQN3 126568894 EC50 = 97 nM T10822 C5OQD7 126584616 EC50 = 7 nM T10822 CZ2U3H 126584619 EC50 = 5.5 nM T10822 CEFR41 126584623 EC50 = 130 nM T10822 COF75Z 126970673 IC50 = 810 nM T10822 C7UN2Q 127030505 IC50 > 10000 nM T10822 CC9X6T 127031177 IC50 = 200 nM T10822 C6CW4R 127031446 IC50 = 56 nM T10822 C5J7YU 127032020 IC50 = 11 nM T10822 C6B8YZ 127034165 IC50 > 30000 nM T10822 CZ1H6I 127034391 IC50 = 18 nM T10822 C9KD6S 127043472 IC50 = 2554 nM T10822 CBQ9G2 127044488 IC50 = 1232 nM T10822 CUH24K 127045941 IC50 = 10.4 nM T10822 CCQR31 127045942 IC50 = 3.3 nM T10822 CN16YJ 127046087 IC50 = 37.4 nM T10822 C4JYB8 127046088 IC50 = 702 nM T10822 C82FLW 127046293 IC50 = 141 nM T10822 C9U1AC 127046294 IC50 = 146 nM T10822 CP9I3G 127046376 IC50 = 2.4 nM T10822 CSL96D 127046538 IC50 = 2.4 nM T10822 CM76FZ 127046539 IC50 = 3.7 nM T10822 C5TJ0Z 127046541 IC50 = 555 nM T10822 CCO3W0 127046703 IC50 = 28 nM T10822 C2ZT5H 127046704 IC50 = 26.9 nM T10822 C56WRF 127047184 IC50 = 10.8 nM T10822 C6EGB3 127047300 IC50 = 14.2 nM T10822 CH3R9M 127047427 IC50 = 5.7 nM T10822 CJV23R 127047567 IC50 = 54.1 nM T10822 CH06YM 127047679 IC50 = 79.3 nM T10822 C58GJF 127047942 IC50 = 47 nM T10822 CDJQ32 127051599 IC50 = 42 nM T10822 C9D1KZ 130423545 IC50 = 2 nM T10822 CD0V7Q 134139422 IC50 > 10000 nM T10822 C1SA4I 134141248 IC50 = 100 nM T10822 CAG82L 134144159 IC50 = 150 nM T10822 C67CQL 134147560 IC50 = 90 nM T10822 CVRB59 134149698 IC50 = 70 nM T10822 C19HTX 134150024 IC50 = 1600 nM T10822 C92PAO 137062026 EC50 = 337 nM T10822 CI1E8V 137634241 IC50 > 10000 nM T10822 CM0UA4 137660456 EC50 > 10000 nM T10822 C9F7IC 138453479 IC50 = 1010 nM T10822 CG1IZ0 145708490 IC50 = 159 nM T10822 CY18FJ 145950114 IC50 = 108 nM T10822 CY3W8C 145950417 IC50 = 24 nM T10822 CTAE93 145950471 IC50 = 34 nM T10822 CG2D9M 145951944 IC50 = 682 nM T10822 CN05WY 145952093 IC50 = 48 nM T10822 CVD80U 145952653 IC50 = 2300 nM T10822 C9X5KZ 145953392 IC50 = 10000 nM T10822 CP1VI4 145954122 IC50 = 10000 nM T10822 C0BU2E 145954767 IC50 = 16 nM T10822 C8TJ0E 145955173 IC50 = 8240 nM T10822 C3P7IZ 145955373 IC50 = 1520 nM T10822 C9V1EY 145955786 IC50 = 208 nM T10822 C8PAW1 145956075 IC50 = 192 nM T10822 C7UI8L 145956330 IC50 = 6000 nM T10822 C4EAX7 145957887 IC50 = 120 nM T10822 C9QTA5 145957989 IC50 = 17 nM T10822 C6P7LD 145958492 IC50 = 24 nM T10822 CPS23D 145958798 IC50 = 443 nM T10822 CZXC30 145959531 IC50 = 1320 nM T10822 CE8X5B 145959610 IC50 = 64 nM T10822 CB6Y3I 145960799 IC50 = 10000 nM T10822 CNM0S5 145961407 IC50 = 164 nM T10822 CN0WS6 145962937 IC50 = 10000 nM T10822 C3P2JL 145970904 IC50 = 17.4 nM T10822 CW4HK8 145975477 IC50 = 10000 nM T10822 CNM5F8 145977216 IC50 = 10000 nM T10822 D01MNK 25125014 IC50 = 90 nM T10822 D0Y2ZC 68115559 IC50 = 22 nM T56108 C36LBD 1250430 IC50 = 9300 nM T56108 C2M0SE 1511198 IC50 > 100000 nM T56108 CJK1F0 1511199 IC50 > 100000 nM T56108 CQ0L9B 2226360 IC50 = 1700 nM T56108 CZ3Y9X 2972356 IC50 = 6170 nM T56108 CR3SF5 4907545 IC50 > 100000 nM T56108 CWG19Q 4908238 IC50 > 100000 nM T56108 CDX05K 5305977 IC50 = 4900 nM T56108 C6RDG4 6459094 IC50 = 23000 nM T56108 CW90UN 9398573 IC50 = 8500 nM T56108 C3FX4U 16028135 IC50 = 10000 nM T56108 C6UCF5 16826960 IC50 = 2500 nM T56108 CIZS84 40889564 IC50 = 3700 nM T56108 C32FNQ 49190359 IC50 = 4000 nM T56108 CTU52G 49190366 IC50 > 10000 nM T56108 CM6Y4O 49190451 IC50 = 3450 nM T56108 CIS4D7 49190466 IC50 > 10000 nM T56108 CDQ80N 50796602 IC50 = 730 nM T56108 CYP58I 50796734 IC50 = 1560 nM T56108 CX12UC 50796762 IC50 = 480 nM T56108 C2GP8Q 50796763 IC50 = 4770 nM T56108 C5UQ8O 50796790 IC50 = 740 nM T56108 CP1U8X 50796792 IC50 = 1470 nM T56108 C1R7BG 50796818 IC50 = 8400 nM T56108 CT34KZ 50796842 IC50 = 2450 nM T56108 CTSH48 50796873 IC50 = 3420 nM T56108 CA01UQ 50796897 IC50 = 2700 nM T56108 CPZ93K 50820616 IC50 = 2700 nM T56108 CA2MT4 50820637 IC50 = 770 nM T56108 CVG1Y0 50820716 IC50 = 1270 nM T56108 CG3PR6 52912222 IC50 = 10000 nM T56108 CIPN50 71760902 IC50 > 10000 nM T56108 C5TB9S 77843982 IC50 > 10000 nM T56108 COZ8S1 78319129 IC50 = 10000 nM T56108 C5NUZ2 91808036 IC50 = 140 nM T56108 CUS7Y0 91808037 IC50 = 57 nM T56108 C7R0MQ 91808039 IC50 = 7.6 nM T56108 CR49YC 118896376 EC50 = 170 nM T56108 C0PY8Z 118896387 EC50 = 120 nM T56108 CM80XC 118896409 EC50 = 2700 nM T56108 CI81CR 118896423 EC50 = 6200 nM T56108 CB74KG 118896464 EC50 = 5000 nM T56108 C5ED8S 118896472 EC50 = 170 nM T56108 CJK35P 118896484 IC50 = 160 nM T56108 C3BY0Z 118896486 EC50 = 59 nM T56108 CP6JD0 118896487 EC50 = 1900 nM T56108 CH3Y4Z 118896503 IC50 = 270 nM T56108 CW29OE 118896529 IC50 = 13 nM T56108 CV0UI6 118896579 EC50 = 110 nM T56108 CUYC60 118896640 IC50 = 60 nM T56108 C4ZK2X 118896672 EC50 = 2300 nM T56108 CL1YV2 118896759 EC50 = 950 nM T56108 C0YR5E 118896778 IC50 = 43 nM T56108 CH04AJ 118909783 IC50 = 160 nM T56108 CUWX94 119081692 IC50 = 910 nM T56108 CZ8S4U 127025422 IC50 = 3690 nM T56108 CB3RH7 127025423 IC50 > 10000 nM T56108 C6TY8H 127025698 IC50 = 4630 nM T56108 CTX9Y6 127029368 IC50 = 2620 nM T56108 CT93VU 127029369 IC50 = 2380 nM T56108 CFH9G7 127029370 IC50 > 10000 nM T56108 C4N6UW 127030551 IC50 = 17000 nM T56108 C70CNT 127030552 IC50 = 4800 nM T56108 C5YPO7 127030561 IC50 = 270 nM T56108 CCF40N 127030853 IC50 = 2800 nM T56108 C8HKB0 127030854 IC50 = 36000 nM T56108 CSL2K3 127031136 IC50 = 14000 nM T56108 CVJ3M7 127031786 IC50 = 2400 nM T56108 C7I9GY 127033003 IC50 = 2000 nM T56108 C8ZQ2U 141736359 IC50 > 20000 nM T56108 C5VNM4 141736367 IC50 > 20000 nM T56108 C96NCH 145950955 IC50 > 20000 nM T56108 C3ZV1O 145952497 IC50 > 20000 nM T56108 CTE74G 145954441 IC50 > 20000 nM T56108 CN5YO3 145957310 IC50 > 20000 nM T56108 C7C5WL 145958595 IC50 = 10440 nM T56108 D03XXT 72201027 IC50 > 20000 nM T56108 D0C2PD 50796983 IC50 = 430 nM T56108 D0O6XT 91827373 IC50 = 1600 nM T80959 D0A7MY 637568 EC50 = 5110 nM T80959 C2UAY1 10455 IC50 > 100000 nM T80959 CKT98D 206035 IC50 > 100000 nM T80959 C9LYF4 286388 IC50 > 25000 nM T80959 CHCF90 665797 IC50 = 3000 nM T80959 CUHT06 899644 IC50 > 25000 nM T80959 CR5D2O 1070170 IC50 > 100000 nM T80959 COY71L 1073725 IC50 = 1800 nM T80959 CAP82W 1103353 IC50 > 25000 nM T80959 CG6UE9 1358452 IC50 = 2800 nM T80959 C60USN 1367926 IC50 > 25000 nM T80959 C9BPG3 1381629 IC50 = 890 nM T80959 CI5C4F 2133805 EC50 = 2900 nM T80959 CL8I0S 2772227 IC50 > 100000 nM T80959 C45EWL 3307826 EC50 > 100000 nM T80959 CXP4D9 6875758 EC50 = 9800 nM T80959 CCDG85 7514662 EC50 = 1120 nM T80959 C7GXT1 8814789 EC50 = 1060 nM T80959 CE2H5T 8814806 EC50 = 1770 nM T80959 CAH31D 8827213 EC50 = 1460 nM T80959 C4PX7O 9815648 IC50 > 100000 nM T80959 CHEX59 10329524 IC50 > 100000 nM T80959 CU79FN 16328219 EC50 = 1460 nM T80959 C1KP4N 40482356 IC50 = 2300 nM T80959 C8FD7E 40482358 EC50 > 100000 nM T80959 CZQ64N 44787480 IC50 > 25000 nM T80959 C8Z3UM 45040448 IC50 > 100000 nM T80959 C3EW7A 50744391 EC50 = 118000 nM T80959 C7PZ9N 56840728 EC50 = 2300 nM T80959 CYVK20 60149024 IC50 = 50118.72 nM T80959 C5HC3B 71681615 IC50 = 22 nM T80959 C3FVN4 71772353 IC50 > 100000 nM T80959 CK3SA1 71812184 EC50 = 1360 nM T80959 C6KD9Z 72189661 EC50 = 2420 nM T80959 C8IB1P 72189966 EC50 = 1630 nM T80959 C1LT8Q 72189968 EC50 = 2060 nM T80959 CS4QL7 72189970 EC50 = 2430 nM T80959 CAN4Z5 72771091 IC50 = 7400 nM T80959 CP7H8X 72771092 IC50 = 750 nM T80959 C38YIA 72771096 IC50 = 1100 nM T80959 C4O1IR 73330369 IC50 = 29 nM T80959 C82RVX 75202265 IC50 > 100000 nM T80959 CH9R1G 77461035 EC50 = 28.6 nM T80959 CBR20Z 91885637 IC50 = 63 nM T80959 CZ8YW7 96002439 EC50 = 5000 nM T80959 CXR0O8 106325804 IC50 > 100000 nM T80959 CXD39Z 118170767 EC50 = 12 nM T80959 C58FEG 118735935 IC50 = 750 nM T80959 CY3QN9 119057445 IC50 = 6200 nM T80959 C1U5AZ 122184660 IC50 = 980 nM T80959 CWY1V7 122184773 IC50 = 966 nM T80959 C1KQ4F 122184774 IC50 = 1666 nM T80959 CBS41H 122184775 IC50 = 10170 nM T80959 C60DTL 122184776 IC50 = 602 nM T80959 C2LR8K 122184777 IC50 = 18.1 nM T80959 C21HBC 122184778 IC50 = 54.3 nM T80959 CI2EZ4 122184779 IC50 = 42.3 nM T80959 CJ07IS 122184780 IC50 = 36.5 nM T80959 CF2MP3 122184781 IC50 = 14.4 nM T80959 CA2T7W 122184782 IC50 = 50.2 nM T80959 CP5NL4 122184783 IC50 = 979 nM T80959 C0OT6L 122184784 IC50 = 34.3 nM T80959 C1MG4H 122184785 IC50 = 179 nM T80959 C47JOU 122184786 IC50 = 47.4 nM T80959 CB9WT4 122184787 IC50 = 122 nM T80959 C1ISB2 122184788 IC50 = 66.1 nM T80959 CR4W6T 122184789 IC50 = 118 nM T80959 CHXM60 122184790 IC50 = 42.2 nM T80959 CL4WB3 122184791 IC50 = 1860 nM T80959 CP9N7W 122190547 EC50 = 5400 nM T80959 CKX08N 122190548 EC50 = 17100 nM T80959 CZL7X3 122190554 EC50 = 11500 nM T80959 CADN59 122190579 EC50 = 20600 nM T80959 C8FU3D 122190580 EC50 = 10000 nM T80959 C1B9FH 122190581 EC50 = 37800 nM T80959 CHS9C4 122190582 EC50 = 22600 nM T80959 C1IXV8 122190583 EC50 = 15000 nM T80959 CR48TK 122190584 EC50 = 11300 nM T80959 C1ID6T 122190585 EC50 = 15000 nM T80959 C96VNR 122190586 EC50 = 38500 nM T80959 C6UNI5 122190587 EC50 = 12700 nM T80959 CMCH49 122190589 EC50 = 8800 nM T80959 C4VK5C 122190590 EC50 = 24500 nM T80959 COC0V8 122190591 EC50 = 7100 nM T80959 C9G2JO 122194678 IC50 = 630 nM T80959 C3TG7O 122194679 IC50 > 25000 nM T80959 C4G5CV 122194680 IC50 > 25000 nM T80959 CPN19J 122194681 IC50 = 1100 nM T80959 CKT2A0 122194682 IC50 = 190 nM T80959 C4U7RN 122194683 IC50 = 660 nM T80959 CE45IP 122194684 IC50 > 25000 nM T80959 C2P8GB 122194685 IC50 > 25000 nM T80959 CA06HT 122194686 IC50 > 25000 nM T80959 CEI45M 122194687 IC50 > 25000 nM T80959 CNOL81 122194688 IC50 > 25000 nM T80959 CQ7NK0 122194689 IC50 > 25000 nM T80959 C9B5FT 122194690 IC50 > 25000 nM T80959 C5D3PT 122194808 IC50 > 25000 nM T80959 CJ28CN 122194809 IC50 = 410 nM T80959 C4KPW8 122194810 IC50 = 85 nM T80959 CLX1H2 122194811 IC50 > 25000 nM T80959 CB7DW0 122194812 IC50 > 25000 nM T80959 C5WZ9F 122194813 IC50 > 25000 nM T80959 CCVQ94 122194814 IC50 > 25000 nM T80959 CT0Q6I 122194815 IC50 = 5500 nM T80959 CGPU04 122194816 IC50 > 25000 nM T80959 C2RUM6 122194817 IC50 > 25000 nM T80959 C6H8SZ 126754132 IC50 < 10 nM T80959 CVL17P 134135178 IC50 = 320 nM T80959 C8IN5B 134139769 IC50 = 875 nM T80959 CLAP94 134141598 IC50 = 200 nM T80959 C9KCA0 134141909 IC50 = 230 nM T80959 CE8SA7 134145193 IC50 = 720 nM T80959 CT62RW 134148665 IC50 = 1300 nM T80959 CSW15J 134150874 IC50 = 634 nM T80959 C28GDW 134152173 IC50 = 3200 nM T80959 CU75YM 134155904 IC50 = 150 nM T80959 C0AG9Z 134813907 IC50 = 60 nM T80959 C85BCI 145951631 IC50 = 1100 nM T80959 CWKC32 145951903 IC50 > 25000 nM T80959 CJPS35 145952403 IC50 > 25000 nM T80959 C4XK3E 145952882 IC50 > 25000 nM T80959 C9N2PW 145952907 IC50 = 101 nM T80959 CIR3D0 145954661 IC50 = 1300 nM T80959 CR67LU 145955145 IC50 = 69700 nM T80959 CW3F9D 145956525 IC50 > 25000 nM T80959 C6UI5X 145956930 IC50 > 25000 nM T80959 CLG56Z 145957104 IC50 > 25000 nM T80959 C0T7QR 145971211 IC50 > 25000 nM T80959 CXLJ15 145973160 IC50 > 25000 nM T80959 CHO10Y 145974303 IC50 > 100000 nM T80959 C5OL0F 145975241 EC50 = 79 nM T80959 CD6L1Q 145979081 IC50 > 100000 nM T80959 CY6PF7 146680922 IC50 = 15.8 nM T80959 CJG46A 155510853 IC50 = 63095.73 nM T80959 C9VYG6 155511125 IC50 > 100000 nM T80959 CUY3M5 155511349 IC50 > 100000 nM T80959 CR01LK 155513180 IC50 = 50118.72 nM T80959 C7ON3W 155513257 IC50 = 19952.62 nM T80959 CK0R4I 155514102 IC50 > 100000 nM T80959 CJ3WP0 155514543 EC50 = 1390 nM T80959 CO9RY3 155515282 IC50 = 50118.72 nM T80959 CUT94K 155515491 EC50 = 970 nM T80959 CTJ97K 155516643 IC50 > 100000 nM T80959 CT28RK 155516991 IC50 = 39810.72 nM T80959 CC9K7R 155517070 IC50 = 50118.72 nM T80959 CYD95J 155517097 IC50 = 39810.72 nM T80959 CP68KM 155517263 IC50 = 50118.72 nM T80959 CB9MT8 155519311 IC50 = 15848.93 nM T80959 C68RTM 155519428 EC50 = 1360 nM T80959 CE6S0K 155519779 IC50 = 6309.57 nM T80959 C9TFN3 155520145 IC50 = 50118.72 nM T80959 C7PO4L 155520368 EC50 = 1910 nM T80959 CYX39S 155520897 EC50 = 1100 nM T80959 CUWL37 155521263 EC50 = 990 nM T80959 CA8IS0 155521928 IC50 = 19952.62 nM T80959 CL65ZK 155524194 IC50 > 100000 nM T80959 CS0WI3 155525300 IC50 = 2600 nM T80959 C73KQP 155525472 IC50 = 39810.72 nM T80959 C3MDZ4 155525522 IC50 > 100000 nM T80959 C4BAY9 155526259 IC50 > 100000 nM T80959 C8JU0Y 155526260 IC50 > 100000 nM T80959 C5RPQ3 155526688 IC50 > 100000 nM T80959 CJX51W 155527016 IC50 > 100000 nM T80959 C90REN 155527528 EC50 = 630 nM T80959 CEP71W 155528033 IC50 = 5011.87 nM T80959 CWI4Q5 155528195 IC50 = 50118.72 nM T80959 CCE2M5 155528362 IC50 > 100000 nM T80959 CS3QI5 155528453 EC50 = 3330 nM T80959 CFO37K 155528822 IC50 = 15848.93 nM T80959 C7L6CB 155529157 IC50 = 12589.25 nM T80959 C38UVP 155529704 IC50 = 12589.25 nM T80959 CKGA51 155530132 IC50 > 100000 nM T80959 C1ZTY3 155530152 IC50 = 63095.73 nM T80959 CEJQ10 155530334 IC50 = 3981.07 nM T80959 CQ4OC5 155531518 IC50 > 100000 nM T80959 CD5B4Z 155531917 IC50 > 100000 nM T80959 CCZ13G 155532065 IC50 = 50118.72 nM T80959 CU1A8Y 155532391 IC50 > 100000 nM T80959 C23ISL 155533277 EC50 = 1230 nM T80959 C7Q8UV 155533600 EC50 = 1540 nM T80959 CPH14B 155533997 IC50 > 50000 nM T80959 C2ZX3Y 155534140 EC50 = 2580 nM T80959 CWQ8P2 155534356 EC50 > 5000 nM T80959 C3K4EL 155535225 IC50 = 5011.87 nM T80959 C0Y9OK 155536020 IC50 = 39810.72 nM T80959 CF36VE 155536250 IC50 = 31622.78 nM T80959 COZC62 155536474 IC50 = 15848.93 nM T80959 CC64FE 155536577 IC50 = 50118.72 nM T80959 CO6ER7 155537046 IC50 = 25118.86 nM T80959 CW7AK4 155537439 IC50 = 15848.93 nM T80959 CK62ID 155537869 IC50 > 100000 nM T80959 C3WE9N 155538368 IC50 = 31622.78 nM T80959 C2RS7E 155539746 IC50 = 609 nM T80959 C75KYA 155540072 IC50 = 19952.62 nM T80959 C6PTE5 155540447 IC50 = 10000 nM T80959 CF0RT5 155540699 IC50 > 100000 nM T80959 CPFC16 155540797 IC50 = 63095.73 nM T80959 C67XKR 155541172 IC50 = 50118.72 nM T80959 C1L0WK 155541675 IC50 > 100000 nM T80959 C43NZV 155542200 IC50 = 10000 nM T80959 CQ8PW0 155542328 IC50 > 100000 nM T80959 CF2P7M 155542638 IC50 > 100000 nM T80959 C4MOF9 155543478 IC50 > 100000 nM T80959 CX8YP9 155543849 EC50 > 5000 nM T80959 C4G6RN 155544017 EC50 > 1000 nM T80959 C2M7EI 155544159 IC50 = 25118.86 nM T80959 C6JOP4 155545387 IC50 = 5011.87 nM T80959 C7UD2J 155546696 IC50 = 50118.72 nM T80959 CZ0I1S 155547074 IC50 > 100000 nM T80959 CQBT74 155547935 IC50 = 19952.62 nM T80959 CO7G5S 155548430 IC50 > 100000 nM T80959 C5XD8R 155548655 IC50 > 100000 nM T80959 C1V5OY 155548738 EC50 = 5520 nM T80959 CEPW05 155549226 IC50 = 100000 nM T80959 CT20GV 155549977 IC50 = 10000 nM T80959 CV4PU6 155550024 IC50 > 50000 nM T80959 CQ1TK8 155550838 EC50 = 1720 nM T80959 C5L8JE 155552136 IC50 > 100000 nM T80959 C9P1KN 155552525 IC50 > 50000 nM T80959 CDK9G7 155553288 IC50 = 2511.89 nM T80959 CH4G2N 155553767 IC50 > 100000 nM T80959 C8YIK6 155553920 IC50 = 25118.86 nM T80959 CNS6W1 155554404 EC50 = 1800 nM T80959 CBQ1U7 155554694 EC50 = 6970 nM T80959 CX83BF 155555686 IC50 = 39810.72 nM T80959 C6WPD1 155555697 IC50 = 50118.72 nM T80959 C0BPZ3 155555710 IC50 = 7943.28 nM T80959 C93OHG 155556364 IC50 = 31622.78 nM T80959 C8BQE6 155556461 IC50 = 15848.93 nM T80959 CQS7P0 155557407 IC50 = 39810.72 nM T80959 CB8Q5Y 155557794 IC50 = 12589.25 nM T80959 CL9F3S 155557868 IC50 = 25118.86 nM T80959 CRL16T 155558461 IC50 = 39810.72 nM T80959 C9XCN2 155558691 IC50 = 31622.78 nM T80959 C1C0ZO 155560119 EC50 = 2840 nM T80959 C24WDN 155560460 IC50 > 100000 nM T80959 CP2H0X 155560853 IC50 > 100000 nM T80959 CB63KG 155561425 IC50 > 100000 nM T80959 CEY87B 155562396 IC50 > 50000 nM T80959 CIJ0H9 155562696 IC50 > 100000 nM T80959 CB6NP3 155563580 IC50 = 31622.78 nM T80959 C13OYN 155563808 IC50 = 31622.78 nM T80959 CP61RM 155564286 IC50 = 31622.78 nM T80959 CA1K9B 155564526 IC50 = 7943.28 nM T80959 C4AL7M 155564597 IC50 > 100000 nM T80959 C85CMZ 155564705 IC50 = 25118.86 nM T80959 C1GUE5 155564896 EC50 = 2300 nM T80959 C6O4NA 155566445 IC50 = 25118.86 nM T80959 CF32ZO 155566614 IC50 > 100000 nM T80959 CC1H8N 155569160 IC50 > 50000 nM T80959 C5P6OE 155569644 IC50 > 100000 nM T80959 D0X4IO 5350 EC50 = 870 nM T05387 D01CCT 25015312 Ki = 1000 nM T05387 D02LBZ 1150683 IC50 = 250 nM T05387 D0CL1D 16094738 Ki = 4000 nM T05387 D0G0EG 3604365 Ki = 15000 nM T05387 D0J4IP 11433028 IC50 = 10000 nM T05387 D0L7MP 54584758 IC50 = 740 nM T05387 D0RX6D 54586674 IC50 = 800 nM T05387 D0UR1H 71459385 IC50 = 62 nM T05387 C4IU5T 6889 IC50 = 65000 nM T05387 C97TNH 10177 IC50 > 100000 nM T05387 C32RNA 82197 IC50 = 58000 nM T05387 C4WEF5 82198 IC50 = 670 nM T05387 C0EH3Z 88695 IC50 = 65000 nM T05387 CJI72V 164610 IC50 = 8000 nM T05387 CC4YZ0 221792 IC50 = 43000 nM T05387 CKTF31 263608 IC50 = 45000 nM T05387 CZT8Q4 263609 IC50 = 3300 nM T05387 C94JHB 346184 IC50 > 80000 nM T05387 CH6W9V 725903 Ki = 10000 nM T05387 CHX80I 906558 IC50 = 25 nM T05387 C9QY6A 1247468 IC50 = 8900 nM T05387 CN42PA 1911570 Ki = 11000 nM T05387 C0WP9N 1970572 IC50 = 30000 nM T05387 CI5K3W 3114310 Ki = 10000 nM T05387 CGR0C9 3250203 IC50 = 29000 nM T05387 CIH3R8 3798517 IC50 > 250000 nM T05387 CD0LT6 5210972 Ki = 3000 nM T05387 C47KRV 5387156 Ki = 4000 nM T05387 CH1Q3A 5858472 IC50 > 2000000 nM T05387 CZ5N4R 6020915 IC50 = 266000 nM T05387 CH7B3C 6179219 IC50 = 688000 nM T05387 CGD0T7 6736443 IC50 > 80000 nM T05387 CC7Y3P 8854099 IC50 = 484000 nM T05387 C8J3CW 10475543 Ki = 48100 nM T05387 CI4JX6 11495693 IC50 > 20000 nM T05387 C07GUF 11502420 IC50 = 480 nM T05387 CT2SY5 11512486 Ki = 34000 nM T05387 CL85JS 11512608 Ki = 51000 nM T05387 C7PY5Z 11516667 IC50 = 3700 nM T05387 CME5G3 11517809 IC50 > 20000 nM T05387 CGT0C2 11526422 Ki = 99000 nM T05387 C5LU8W 11532188 IC50 = 1300 nM T05387 CX69AW 11538401 IC50 = 230 nM T05387 C0WO3S 11539509 IC50 = 1500 nM T05387 CB4D5I 11604719 IC50 > 20000 nM T05387 C4ZT6Y 11606581 Ki = 18000 nM T05387 C95JGH 11620297 Ki = 22000 nM T05387 C4WHA7 11626706 Ki = 138000 nM T05387 CY7G4M 11632564 IC50 = 4500 nM T05387 CJ9C7B 11633193 IC50 > 10000 nM T05387 CIH4U0 11633950 IC50 > 20000 nM T05387 C2NS1P 11642087 Ki = 19000 nM T05387 CU0S1P 11647123 IC50 > 20000 nM T05387 C26QZE 11655066 IC50 = 2100 nM T05387 C2CH9V 11662546 IC50 > 20000 nM T05387 CV4K5X 11677975 Ki = 18000 nM T05387 CPD35K 11784890 IC50 = 130 nM T05387 CZD2M4 12192833 IC50 = 3800 nM T05387 CM1VP7 12214258 IC50 = 18000 nM T05387 CSB6W1 13593050 IC50 > 80000 nM T05387 CK2NL0 14159824 Ki = 68000 nM T05387 C6JIA9 14977359 IC50 = 1001000 nM T05387 C9XY0T 16094735 Ki = 41000 nM T05387 CT0J2Q 16094739 Ki = 30000 nM T05387 CK9QS3 16094740 Ki = 1300 nM T05387 C16GQH 16094746 Ki = 62000 nM T05387 CMFB75 16094751 Ki = 11000 nM T05387 CDO05F 16794671 IC50 = 65000 nM T05387 C50DXP 17578027 IC50 = 8500 nM T05387 C1UH6R 21657832 IC50 = 3000 nM T05387 C93LAQ 28254071 IC50 = 160 nM T05387 CGYM83 43405474 IC50 = 1900 nM T05387 C48LFD 43616300 IC50 = 26000 nM T05387 C35YMI 43616336 IC50 = 5000 nM T05387 CB15SK 44177708 IC50 = 30 nM T05387 CK61PE 44391413 IC50 = 140 nM T05387 CF56IQ 44391417 IC50 = 1500 nM T05387 C2A9MD 44391420 IC50 = 5300 nM T05387 CF6RG7 44391421 IC50 = 1800 nM T05387 C6TWE1 44391422 IC50 = 160 nM T05387 CB49WR 44391423 IC50 = 140 nM T05387 CC6BL9 44391427 IC50 = 170 nM T05387 C35RQG 44391432 IC50 = 8400 nM T05387 C9E8RC 44391436 IC50 = 2300 nM T05387 CTZS65 44391437 IC50 = 150 nM T05387 CN6PF9 44391438 IC50 = 180 nM T05387 CHN67G 44391439 IC50 = 320 nM T05387 CF8JC0 44391442 IC50 = 2300 nM T05387 CI05BQ 44391446 IC50 = 1400 nM T05387 CV28CQ 44391447 IC50 = 2600 nM T05387 C1IJX6 44391448 IC50 = 6300 nM T05387 CWA98E 44391451 IC50 = 4800 nM T05387 C0Y2NA 44391453 IC50 = 2000 nM T05387 CE20LY 44391454 IC50 = 1100 nM T05387 C6CKW3 44391456 IC50 = 820 nM T05387 C4G7JH 44391457 IC50 = 900 nM T05387 CT1S3I 44391463 IC50 = 280 nM T05387 C8SA0H 44391464 IC50 = 290 nM T05387 CE35YW 44391465 IC50 = 290 nM T05387 C58DZS 44391466 IC50 > 20000 nM T05387 C4XW1Z 44391467 IC50 = 7100 nM T05387 CZY68W 44391468 IC50 = 530 nM T05387 C0EUL6 44391472 IC50 = 450 nM T05387 C8SGD0 44391479 IC50 > 20000 nM T05387 CMS98F 44391481 IC50 > 20000 nM T05387 CX9KC0 44391482 IC50 = 140 nM T05387 C5HKO4 44391483 IC50 = 1800 nM T05387 CITE65 44391484 IC50 = 6000 nM T05387 C20HKU 44391489 IC50 = 200 nM T05387 CK1Y8S 44437812 Ki = 300000 nM T05387 CZ4T9V 44437813 Ki = 40000 nM T05387 CV3YP9 44437814 Ki = 200000 nM T05387 CF8R4L 44589634 IC50 = 20000 nM T05387 C5KSW0 44589636 IC50 = 3000 nM T05387 CZ3LE4 44590162 IC50 = 8000 nM T05387 C9H5JS 51039927 IC50 = 10 nM T05387 CHT9R4 52938041 IC50 = 46 nM T05387 C0ON6R 52938045 IC50 = 44 nM T05387 C9H5GZ 52938046 IC50 = 37 nM T05387 CEV19T 52938170 IC50 = 57 nM T05387 CF59EP 52938291 IC50 = 380 nM T05387 C08STG 52938293 IC50 = 78 nM T05387 C6YOG9 52938294 IC50 = 310 nM T05387 CY5VE4 52938668 IC50 = 110 nM T05387 CH9X0Y 52938669 IC50 = 32 nM T05387 C3ELI5 52938797 IC50 = 810 nM T05387 CVH6P1 52939047 IC50 = 97 nM T05387 CW4A3I 52939048 IC50 = 140 nM T05387 C9G3TL 52939163 IC50 = 54 nM T05387 CMU46C 52939516 IC50 = 120 nM T05387 C4OK5Z 52939517 IC50 = 350 nM T05387 CNJ3E5 52939518 IC50 = 460 nM T05387 CM0B1P 52939519 IC50 = 120 nM T05387 CL1C8U 52939520 IC50 = 450 nM T05387 CV67SO 52939643 IC50 = 220 nM T05387 C4NY5P 52939644 IC50 = 94 nM T05387 C7X1PB 52939647 IC50 = 96 nM T05387 CHGK38 52939771 IC50 = 180 nM T05387 C0F5JG 52939772 IC50 = 1500 nM T05387 CLF5S8 52939773 IC50 = 380 nM T05387 C3H8EG 52939774 IC50 = 210 nM T05387 CG49TO 52939776 IC50 = 110 nM T05387 CTCF48 52939902 IC50 = 500 nM T05387 CWOX98 53359813 IC50 = 180 nM T05387 C6IQJ4 54580777 Ki = 900 nM T05387 C32LVS 54580801 Ki = 4000 nM T05387 C05ACQ 54580802 IC50 = 660 nM T05387 CUCO54 54581832 IC50 = 1400 nM T05387 C6VI1F 54581833 IC50 = 2900 nM T05387 CE36RP 54581834 IC50 = 1000 nM T05387 CYXC46 54581835 IC50 = 5500 nM T05387 CG4VM2 54581836 IC50 = 6300 nM T05387 CKG0Y4 54581837 IC50 = 360 nM T05387 C08WHD 54582753 Ki = 700 nM T05387 CY7IZ9 54582754 IC50 = 1100 nM T05387 CHD18E 54582755 IC50 = 1200 nM T05387 C6B0YU 54582781 IC50 = 1400 nM T05387 CNHJ27 54582782 IC50 = 1200 nM T05387 C1TRB9 54583744 IC50 = 3900 nM T05387 C01YHW 54583769 IC50 = 1100 nM T05387 CVQ75I 54583770 IC50 = 360 nM T05387 CW1Q2L 54583771 IC50 = 560 nM T05387 CLBA79 54584722 Ki = 5400 nM T05387 C24DIA 54584723 IC50 = 2600 nM T05387 CPKC63 54584756 Ki = 3300 nM T05387 CD1RL3 54584757 IC50 = 90 nM T05387 CF9PZ1 54584759 Ki = 250 nM T05387 CIA6G0 54584760 IC50 = 2100 nM T05387 C9E1MU 54585611 IC50 = 900 nM T05387 CGF9X8 54585688 IC50 = 700 nM T05387 CUH0G4 54585689 IC50 = 1400 nM T05387 C36QET 54585690 IC50 = 2100 nM T05387 CQJ0F6 54585691 IC50 = 1800 nM T05387 CUS1F0 54585692 IC50 = 1700 nM T05387 CH0YI2 54585693 IC50 = 2900 nM T05387 CY0F4O 54586646 IC50 = 1400 nM T05387 C5GB9Y 54586672 IC50 = 1000 nM T05387 CKF1M2 54586673 IC50 = 1000 nM T05387 CX6BF9 54586675 IC50 = 1100 nM T05387 CG9P1E 54587706 IC50 = 1100 nM T05387 CXMP30 54587707 IC50 = 7300 nM T05387 C5HA4R 56953730 IC50 = 1300 nM T05387 CTMS75 56953731 IC50 = 4500 nM T05387 C7TN6K 56953732 IC50 = 2900 nM T05387 CHNG07 56953735 IC50 = 55 nM T05387 C3Z8BE 56953736 IC50 = 25 nM T05387 CHYL72 56953863 IC50 = 35 nM T05387 C8AY9P 56953864 IC50 = 52 nM T05387 CI6L1M 56953865 IC50 = 76 nM T05387 CB4T3M 56953866 IC50 = 180 nM T05387 CJ4CU6 56953867 IC50 = 190 nM T05387 C14JIX 56953989 IC50 = 580 nM T05387 C3WZA9 56953990 IC50 = 520 nM T05387 C19DEA 56954113 IC50 = 54 nM T05387 C3Q1MG 56954114 IC50 = 70 nM T05387 CZQ09H 56954116 IC50 = 70 nM T05387 CIAL27 56954117 IC50 = 82 nM T05387 CO7WI3 56954118 IC50 = 220 nM T05387 CJ9Z8T 56954217 IC50 = 110 nM T05387 CQP53N 56954218 IC50 = 20 nM T05387 CYV7I4 56954219 IC50 = 26 nM T05387 CF0L3O 56954220 IC50 = 160 nM T05387 CCS1W8 56954302 IC50 = 34 nM T05387 CNL06J 56954305 IC50 = 180 nM T05387 CX89IJ 56954306 IC50 = 15 nM T05387 CYB8K2 56954307 IC50 = 26 nM T05387 C7RS2X 56954413 IC50 = 69 nM T05387 C8HKW1 56954414 IC50 = 14 nM T05387 C2TV9J 56954416 IC50 = 28000 nM T05387 CV2M0I 56954417 IC50 = 2300 nM T05387 CQ9G1B 56954418 IC50 > 80000 nM T05387 CQ06DB 56954502 IC50 = 2800 nM T05387 CK2W7N 56954503 IC50 = 2800 nM T05387 C9L3UE 56954504 IC50 > 80000 nM T05387 C0JM9C 56954505 IC50 > 10000 nM T05387 C68FIA 56954506 IC50 > 10000 nM T05387 CJZ47H 56954507 IC50 = 140 nM T05387 CFI7L9 56954609 IC50 = 6800 nM T05387 CMPI75 56954610 IC50 > 80000 nM T05387 C9ECY6 56954611 IC50 > 80000 nM T05387 C7MBC5 56954612 IC50 > 80000 nM T05387 C53PIX 56954613 IC50 > 80000 nM T05387 CO91HU 56954614 IC50 > 80000 nM T05387 CX3NW5 56954720 IC50 = 1400 nM T05387 C30RHS 56954721 IC50 > 80000 nM T05387 C74KPC 56954722 IC50 = 91000 nM T05387 CL2B8Y 56954825 IC50 = 76000 nM T05387 C8XMJ9 56954826 IC50 = 13000 nM T05387 CZL5M6 56954827 IC50 = 2500 nM T05387 CHA2O7 56954828 IC50 = 910 nM T05387 C3KSN7 56954829 IC50 = 190 nM T05387 CXQG95 56954830 IC50 = 110 nM T05387 C27JWY 56954942 IC50 = 72 nM T05387 CIP9V4 57251115 IC50 = 43000 nM T05387 C02CZV 58435684 IC50 = 54 nM T05387 CMK76O 61113906 IC50 > 80000 nM T05387 CBD36K 70682660 IC50 = 16000 nM T05387 C1M7WL 70687120 IC50 = 300 nM T05387 CNY61X 70688957 IC50 = 130 nM T05387 C38DBS 70691276 IC50 = 30000 nM T05387 C4ZB7K 70693195 IC50 = 60 nM T05387 C1K5WF 70695295 IC50 = 5700 nM T05387 CDS6T7 71096277 IC50 = 20 nM T05387 CWL96G 71449433 IC50 = 280 nM T05387 C31KGX 71449434 IC50 = 5100 nM T05387 CF9XS0 71449435 IC50 > 80000 nM T05387 C9EV4K 71449437 IC50 = 380 nM T05387 CVE80H 71449438 IC50 = 320 nM T05387 C97SYI 71449439 IC50 = 310 nM T05387 CE13PK 71449440 IC50 = 460 nM T05387 C6Z3ES 71449441 IC50 = 180 nM T05387 CPQC71 71450339 IC50 > 80000 nM T05387 C9I4MT 71450340 IC50 = 78 nM T05387 CE7T4G 71450341 IC50 = 55 nM T05387 C31MWX 71450342 IC50 = 160 nM T05387 CR9CK8 71450343 IC50 = 3100 nM T05387 CQR82A 71450344 IC50 = 62000 nM T05387 CS1RH3 71450345 IC50 = 1100 nM T05387 C5DRO4 71451225 IC50 > 80000 nM T05387 CBXQ58 71451226 IC50 = 55000 nM T05387 CUB8Z1 71451230 IC50 = 280 nM T05387 C4FW0X 71451231 IC50 = 170 nM T05387 CYUA29 71452144 IC50 = 190 nM T05387 C3K8UY 71452145 IC50 = 850 nM T05387 CKT15B 71452146 IC50 = 1800 nM T05387 C51IRQ 71452147 IC50 = 730 nM T05387 CPXV51 71452148 IC50 = 230 nM T05387 CBM94I 71452149 IC50 = 7600 nM T05387 CDLT23 71452150 IC50 > 80000 nM T05387 C04ANU 71452151 IC50 = 21000 nM T05387 C4VK1B 71453043 IC50 = 30000 nM T05387 CW2TF6 71453044 IC50 = 770 nM T05387 CGWL48 71453046 IC50 = 550 nM T05387 C1HZ4R 71453047 IC50 = 8900 nM T05387 C6VWS4 71453979 IC50 = 110 nM T05387 C9KJV7 71453980 IC50 = 170 nM T05387 CTYQ16 71453981 IC50 = 7900 nM T05387 CP4B2W 71453982 IC50 = 5900 nM T05387 CP6U7R 71453983 IC50 = 9100 nM T05387 CBJF60 71454785 IC50 = 3300 nM T05387 CW37TL 71454786 IC50 = 630 nM T05387 CYDH61 71454789 IC50 = 660 nM T05387 CP8TF2 71454790 IC50 = 360 nM T05387 C65ZIA 71454791 IC50 = 57000 nM T05387 CMA7K3 71455724 IC50 = 1400 nM T05387 C24YSA 71455725 IC50 = 54 nM T05387 CSXR49 71455726 IC50 = 610 nM T05387 C9T8XL 71455727 IC50 = 3500 nM T05387 CT8G9O 71455728 IC50 = 14000 nM T05387 C87DGK 71456561 IC50 = 1600 nM T05387 CGA32C 71456564 IC50 = 200 nM T05387 CB64IG 71456565 IC50 = 110 nM T05387 CK9HB3 71456566 IC50 = 22000 nM T05387 C1D6LM 71456567 IC50 = 280 nM T05387 C20RDV 71456568 IC50 = 230 nM T05387 CICA80 71457506 IC50 > 80000 nM T05387 CTA97S 71457507 IC50 = 2700 nM T05387 CWD4V2 71457508 IC50 = 33000 nM T05387 CRQL03 71457509 IC50 = 10000 nM T05387 C4LBJ6 71458416 IC50 = 620 nM T05387 C8Y2CE 71458420 IC50 = 1600 nM T05387 C97KNM 71459379 IC50 = 1600 nM T05387 CW7MP0 71459380 IC50 = 1200 nM T05387 CJ31OB 71459381 IC50 = 2500 nM T05387 CS0PX1 71459382 IC50 = 590 nM T05387 C8YF6H 71459383 IC50 = 660 nM T05387 CY0IH6 71459384 IC50 = 240 nM T05387 CV7QI8 71459386 IC50 = 260 nM T05387 CKXS41 71459387 IC50 = 5400 nM T05387 COI05G 71459388 IC50 = 10000 nM T05387 COSL04 71459389 IC50 = 14000 nM T05387 C2BHC5 71460257 IC50 = 200 nM T05387 C5GRH8 71460258 IC50 = 140 nM T05387 CA3VR1 71460263 IC50 = 170 nM T05387 CCR2A7 71460264 IC50 = 280 nM T05387 CI35VO 71461138 IC50 = 1900 nM T05387 C1IV9T 71461964 IC50 = 410 nM T05387 C9DIB0 71461965 IC50 = 460 nM T05387 C4EO3L 71461969 IC50 = 260 nM T05387 CGM68H 71462877 IC50 = 14 nM T05387 C2CG9W 71462878 IC50 = 190 nM T05387 C7T5XI 71462879 IC50 = 580 nM T05387 C62KMF 72204717 IC50 = 1000 nM T05387 CN6D1U 72204898 IC50 > 200000 nM T05387 CG0MH1 72204900 IC50 > 200000 nM T05387 CPN93S 72204902 IC50 > 200000 nM T05387 CIN2X8 72204904 IC50 > 200000 nM T05387 C7P2VY 72205081 IC50 > 200000 nM T05387 C1R6BL 72205083 IC50 > 200000 nM T05387 CI3PV6 72205085 IC50 > 200000 nM T05387 CJA86H 72205087 IC50 > 200000 nM T05387 C8WSG4 72205270 IC50 = 5000 nM T05387 CN52BD 72205272 IC50 = 10000 nM T05387 C93THM 72205274 IC50 = 20000 nM T05387 C5W3HF 72950407 IC50 = 45 nM T05387 CUFW53 73775533 IC50 = 6 nM T05387 CYX2V6 76447116 IC50 = 4000 nM T05387 C3INA2 118736260 IC50 = 150 nM T05387 CNQ12A 118736261 IC50 = 46 nM T05387 CW61EZ 118736262 IC50 = 48 nM T05387 CRT3P7 118736263 IC50 = 50 nM T05387 C7G1DH 118736264 IC50 = 1100 nM T05387 C0Z8VF 118736265 IC50 = 57 nM T05387 C1BQM5 118736266 IC50 = 9.6 nM T05387 CX2Y0R 118736267 IC50 = 130 nM T05387 C02SAE 118736268 IC50 = 88 nM T05387 CF32KR 118736270 IC50 = 48 nM T05387 CGK5M6 118736271 IC50 = 150 nM T05387 C53RDV 121487961 Ki = 13400 nM T05387 CV30MT 121487964 Ki = 11200 nM T05387 CC4BH5 132024475 Ki = 8900 nM T05387 CS68YV 132024504 Ki = 12900 nM T05387 CQ30BT 135403657 Ki = 27000 nM T05387 C5QM1T 136233424 IC50 = 200 nM T05387 C7VDE2 136233425 IC50 = 16000 nM T05387 CJY42A 137632110 Ki = 9100 nM T05387 C4UL1P 137634041 Ki = 38700 nM T05387 CV9MC4 137636961 Ki = 20000 nM T05387 CWR61U 137637535 Ki = 10400 nM T05387 CV40UF 137637578 Ki = 6700 nM T05387 CTG86Z 137638796 Ki = 14700 nM T05387 CB10SH 137640581 Ki = 40000 nM T05387 CV8G9H 137642100 Ki = 36000 nM T05387 C36BWL 137643267 Ki = 47700 nM T05387 CP4LA8 137643826 Ki = 36600 nM T05387 C0YUP8 137645880 Ki = 30500 nM T05387 CH5PC1 137647516 Ki = 8800 nM T05387 CEX3M1 137650985 Ki = 52100 nM T05387 CNS4A6 137651280 Ki = 23500 nM T05387 CZ2IB9 137652230 Ki = 6400 nM T05387 C3J5KW 137655115 Ki = 11000 nM T05387 CT2WY3 137655910 Ki = 35100 nM T05387 C12UCI 137659185 Ki = 32100 nM T05387 C2ALI7 137659798 Ki = 33900 nM T05387 CH8FA4 137659888 Ki = 27100 nM T05387 C9J2LZ 137661143 Ki = 40100 nM T05387 CTF01B 137661324 Ki = 23400 nM T05387 C4RBT0 145951882 IC50 = 151000 nM T05387 C63JGU 145952387 IC50 = 25900 nM T05387 CEF02T 145952817 Ki = 420 nM T05387 C02KYA 145954920 IC50 = 64100 nM T05387 CI14SB 145955271 Ki = 9900 nM T05387 C6DNE2 145955756 IC50 = 147000 nM T05387 CDX14L 145955913 IC50 > 100000 nM T05387 C9CV2F 145957661 IC50 = 2600 nM T05387 CU6W8S 145959648 IC50 > 100000 nM T05387 C60XHM 145960783 IC50 > 100000 nM T05387 C16NDU 145962928 IC50 = 145000 nM T05387 CRZ18N 145967599 Ki = 6770 nM T05387 C7LZA4 145967697 Ki = 64300 nM T05387 CSH74V 145967717 IC50 = 390 nM T05387 C4B2IN 145967901 Ki = 7960 nM T05387 CTO79E 145967965 Ki = 14000 nM T05387 C6HW3T 145968169 Ki = 2600 nM T05387 COVJ90 145968339 Ki = 7710 nM T05387 CR8L5N 145968416 Ki = 7600 nM T05387 CON65L 145968505 Ki = 7120 nM T05387 CPF7K0 145968648 IC50 = 1100 nM T05387 CV3AX6 145968665 Ki = 5560 nM T05387 C18HAN 145968666 IC50 = 170 nM T05387 CD8WE6 145968855 IC50 = 100 nM T05387 C6GTR0 145969042 Ki = 6810 nM T05387 C4YM5Z 145969060 Ki = 10900 nM T05387 CYG97J 145969130 Ki = 5020 nM T05387 CAP4S6 145969324 IC50 = 140 nM T05387 CT3ES8 145969645 Ki = 2520 nM T05387 CHD7X4 145969733 Ki = 4490 nM T05387 CZ0G3Y 145969956 IC50 = 200 nM T05387 C5QVF1 145969982 IC50 = 180 nM T05387 C2PL7F 145970586 Ki = 13400 nM T05387 CN2U3K 145970701 Ki = 14300 nM T05387 CM43US 145970727 IC50 = 220 nM T05387 C87PHO 145971057 Ki = 7550 nM T05387 CA1C4T 145971062 IC50 = 340 nM T05387 C91WUG 145971267 IC50 = 610 nM T05387 CZO4N8 145986797 IC50 = 90 nM T05387 CDEL85 145987285 Ki = 15000 nM T05387 C1ND0C 145987727 Ki = 5720 nM T05387 C9LEF7 145987736 Ki = 2550 nM T05387 CMIV48 145988826 Ki = 1980 nM T05387 D03TPH 87203 IC50 = 65000 nM T05387 D0N6BC 950368 Ki = 100000 nM T05387 D0SP2O 7054 IC50 > 250000 nM T15377 D07SDQ 969516 IC50 = 7000 nM T15377 CIVG56 44140287 Ki = 11 nM T15377 CTA9U7 76900277 Ki = 27 nM T15377 CD6I4N 135494311 IC50 = 90 nM T15377 CQX58A 155539389 Ki = 1.3 nM T15377 C9Y4XJ 155546938 IC50 = 210 nM T15377 D0M5LP 2374 IC50 = 2000 nM T15377 D0V4WT 105008 IC50 = 5000 nM T95761 C8PB3W 25255921 IC50 = 240 nM T95761 C2L6BY 127044673 IC50 = 378 nM T95761 C3U7SO 127044674 IC50 = 452 nM T95761 CMD8X7 127044675 IC50 > 5000 nM T95761 CRN5I8 127044676 IC50 > 5000 nM T95761 C3VN2U 127044838 IC50 = 157 nM T95761 CZIT53 127044839 IC50 = 1645 nM T95761 CK4SN9 127044840 IC50 = 420 nM T95761 C8O1XJ 127044845 IC50 = 2345 nM T95761 CXK9T4 127044846 IC50 = 890 nM T95761 C3P9GU 127045001 IC50 = 192 nM T95761 C1P0IJ 127045002 IC50 = 368 nM T95761 CSR17Z 127045008 IC50 = 256 nM T95761 C9A1IR 127045009 IC50 = 220 nM T95761 C6T8SP 127045153 IC50 = 142 nM T95761 CQ1VL6 127045154 IC50 = 182 nM T95761 CET10Z 127045301 IC50 > 5000 nM T95761 CMJ4X2 127045302 IC50 > 10000 nM T95761 CL84CO 127045303 IC50 = 1245 nM T95761 D06EHW 11625778 IC50 = 1000 nM T53585 D01QIN 60823 IC50 = 6 nM T53585 D02RQU 54687 IC50 = 30 nM T53585 D03KIA 446156 IC50 = 10 nM T53585 D06WTZ 53232 IC50 = 0.05 nM T53585 D0E7PQ 5311 IC50 > 10000 nM T53585 D0G1WL 5282451 IC50 = 8900 nM T53585 D0H0ND 54454 IC50 = 0.9 nM T53585 D0JE2E 446157 Ki = 0.9 nM T53585 D0J9GD 64715 IC50 = 23 nM T53585 D0U5NU 5281970 IC50 = 5 nM T53585 CX5V2H 636822 IC50 = 5860 nM T53585 C0LQ7X 5314397 IC50 = 22.91 nM T53585 CG53MU 5353627 IC50 = 28 nM T53585 CGD21K 6439471 IC50 = 6.15 nM T53585 CRG02H 9865943 IC50 = 18 nM T53585 CNWH06 10065248 IC50 = 10000 nM T53585 CY1EG2 11442745 IC50 = 21700 nM T53585 C9POB8 11753476 IC50 = 1.8 nM T53585 C4TKF1 12306828 IC50 = 8400 nM T53585 C8YBC1 13298846 IC50 = 12.1 nM T53585 COU43B 14460200 IC50 = 2000 nM T53585 CD0OZ5 14460203 IC50 = 5000 nM T53585 C91JPM 14460204 IC50 = 90 nM T53585 C9GXT3 14460209 IC50 = 20 nM T53585 C7OA1K 14460211 IC50 = 9.5 nM T53585 C1M9BO 14460213 IC50 > 5000 nM T53585 CERL21 14460221 IC50 = 5 nM T53585 CJ9O0M 14849847 IC50 = 9 nM T53585 C16DQL 15663484 IC50 = 8 nM T53585 CA67TN 15934934 IC50 = 1700 nM T53585 CZ5V3O 15934936 IC50 = 4900 nM T53585 CLHO84 16759173 IC50 = 30 nM T53585 C61NDV 16760544 IC50 = 29 nM T53585 CW9DF2 16760655 IC50 = 12 nM T53585 C0QWE9 23665944 IC50 = 1340 nM T53585 CIJ2Z0 23688546 IC50 = 59 nM T53585 C98ETA 23695878 IC50 = 8 nM T53585 CL75XP 23695881 IC50 = 66 nM T53585 CX4W6U 23695889 IC50 = 7 nM T53585 CGVR91 23708535 IC50 = 1.8 nM T53585 CKVS96 23708976 IC50 = 16.7 nM T53585 C8N2SU 23714444 IC50 < 0.01 nM T53585 CF53LC 24763877 IC50 = 0.8 nM T53585 C91XJY 24944096 IC50 = 12 nM T53585 C6E1OJ 25166691 IC50 = 75230 nM T53585 CSL3W9 25166692 IC50 = 44810 nM T53585 CW4M9B 25166903 IC50 = 52670 nM T53585 C5TC9D 25166904 IC50 = 41210 nM T53585 C7BE6Y 40785065 IC50 = 2.2 nM T53585 CVT1H2 44224156 IC50 = 30200 nM T53585 C1I3ZF 44267525 IC50 = 1290 nM T53585 C8P0HR 44267551 IC50 = 1720 nM T53585 CTPZ78 44285668 Ki = 3 nM T53585 C12UMX 44306438 IC50 = 40 nM T53585 C4HJ0V 44306551 IC50 = 20 nM T53585 C0D8NG 44306815 IC50 = 110 nM T53585 CHX70L 44331510 IC50 > 5000 nM T53585 CY92SA 44331598 IC50 = 100 nM T53585 C0KMF8 44331627 IC50 = 10000 nM T53585 C30RHG 44331644 IC50 = 12000 nM T53585 C0L2JN 44331886 IC50 = 6500 nM T53585 CK87FH 44331887 IC50 = 2500 nM T53585 C1A0TH 44331896 IC50 > 1700 nM T53585 CI3MJ6 44331955 IC50 > 1000 nM T53585 CE0C2W 44332018 IC50 > 5000 nM T53585 CI94KW 44332020 IC50 = 5.6 nM T53585 C4ET6Z 44332034 IC50 = 55 nM T53585 COL8H4 44332036 IC50 > 500 nM T53585 CXG61C 44332134 IC50 = 20000 nM T53585 CPA40M 44342306 IC50 = 2220 nM T53585 CYG7B1 44346747 IC50 = 7.52 nM T53585 C6P7IL 44347122 IC50 = 8.4 nM T53585 C6R5EK 44347157 IC50 = 7.89 nM T53585 CI91MR 44347309 IC50 = 7.25 nM T53585 CD92JW 44347322 IC50 = 7.66 nM T53585 CG70FO 44347337 IC50 = 8.1 nM T53585 CP74VN 44347339 IC50 = 9 nM T53585 C41RIT 44347341 IC50 = 8.04 nM T53585 CJ1N2T 44347351 IC50 = 8.52 nM T53585 C8VKD3 44347366 IC50 = 8.15 nM T53585 C7K8TP 44347369 IC50 < 7 nM T53585 CZ4IA8 44347391 IC50 = 9 nM T53585 CH9UN3 44347404 IC50 = 8.7 nM T53585 C0OP7R 44347423 IC50 = 8.7 nM T53585 CS21WC 44347427 IC50 = 7 nM T53585 CEAX43 44354271 IC50 = 1500 nM T53585 CL95ZY 44365204 IC50 = 1500000 nM T53585 CJI67T 44365475 IC50 = 4600 nM T53585 C2XN4K 44374858 IC50 = 0.002 nM T53585 C0UPV7 44374900 IC50 = 0.014 nM T53585 C02ILW 44375049 IC50 = 5 nM T53585 CI4M8R 44375051 IC50 = 6 nM T53585 CSI1Q7 44387497 IC50 = 4.1 nM T53585 CCOM85 44392469 IC50 = 9.52 nM T53585 CIC37P 44392485 IC50 = 7.6 nM T53585 C5T2DU 44392493 IC50 = 8.7 nM T53585 C03DYG 44392496 IC50 = 7.15 nM T53585 C1E5HF 44392505 IC50 = 8.7 nM T53585 CGKC06 44392507 IC50 = 7.16 nM T53585 CD1JO0 44392516 IC50 = 9.3 nM T53585 C2Y1CI 44392525 IC50 = 8.3 nM T53585 CWCH72 44392541 IC50 = 8.7 nM T53585 CC0UF3 44426467 IC50 = 9.6 nM T53585 CJ0X8U 44426476 IC50 = 2.9 nM T53585 C3NZ5F 44426479 IC50 = 16.4 nM T53585 CWK87Y 44426482 IC50 = 13.9 nM T53585 C3WR4O 44426484 IC50 = 3 nM T53585 CH7XU1 44426486 IC50 = 37.4 nM T53585 C0P8IG 44426488 IC50 = 4.7 nM T53585 CQ32BZ 44426490 IC50 = 11.7 nM T53585 C8D3YG 44426492 IC50 = 3.5 nM T53585 CY1JN0 44426494 IC50 = 3 nM T53585 C68OPB 44442190 IC50 = 6.6 nM T53585 CKJ6Z2 44442191 IC50 = 12.4 nM T53585 CJF2K5 44442192 IC50 = 0.7 nM T53585 CL9U7E 44442193 IC50 = 0.4 nM T53585 C2UMQ6 44442195 IC50 = 0.3 nM T53585 CGHW16 44442196 IC50 = 0.3 nM T53585 CJQ3C6 44442199 IC50 = 1.4 nM T53585 CBU17T 44442202 IC50 = 2.9 nM T53585 CY5DP8 44442203 IC50 = 0.3 nM T53585 C63PRO 44442205 IC50 = 0.8 nM T53585 C7X2ZO 44442208 IC50 = 0.7 nM T53585 C9W6GZ 44442211 IC50 = 1.8 nM T53585 CN7HT8 44442216 IC50 = 1.2 nM T53585 CUPB61 44442219 IC50 = 1.2 nM T53585 CV54GT 44442221 IC50 = 2.2 nM T53585 CW2CM1 44442223 IC50 = 1.5 nM T53585 CM8VH1 44442226 IC50 = 0.8 nM T53585 CUV4M6 44442232 IC50 = 0.6 nM T53585 C9O0FG 44442237 IC50 = 2.6 nM T53585 C7MWL0 44442240 IC50 = 3.4 nM T53585 CM7DQ0 44442243 IC50 = 3 nM T53585 CHE19M 44442247 IC50 = 8.8 nM T53585 C6Q4WG 44442253 IC50 = 20 nM T53585 CPI23U 44442258 IC50 = 15 nM T53585 CV45BF 44442260 IC50 = 3.8 nM T53585 C6ZA0D 44451948 IC50 = 201120 nM T53585 CPAB62 44451976 IC50 = 484720 nM T53585 CND0U9 44452214 IC50 = 27280 nM T53585 CL2RS9 44584795 IC50 = 60 ug.mL-1 T53585 CLQ6B8 46196547 IC50 = 6930 nM T53585 CIV2D5 46196548 IC50 = 5610 nM T53585 CUV9P0 46196560 IC50 = 7100 nM T53585 CBT1X3 46227441 IC50 = 62400 nM T53585 C4H0ES 46227447 IC50 = 25700 nM T53585 C4EFZ2 46227470 IC50 = 11300 nM T53585 C8FP1N 46227471 IC50 = 41300 nM T53585 CW51NY 46227475 IC50 = 359600 nM T53585 CF62RP 46227476 IC50 = 759000 nM T53585 CEU8O9 46227488 IC50 = 45700 nM T53585 CCA45R 46871863 IC50 = 39.81 nM T53585 CZVF15 46906129 Ki = 260 nM T53585 CMD60F 46906130 IC50 = 6950 nM T53585 CJ6KS2 46906162 IC50 = 2560 nM T53585 C1Z0TF 46906164 IC50 = 410 nM T53585 C4HQR9 46906165 IC50 = 8520 nM T53585 CMF6S7 46906166 IC50 = 270 nM T53585 CWS8T7 46906167 IC50 = 260 nM T53585 C3E1YK 46906169 IC50 = 240 nM T53585 C7EP4L 46906528 IC50 = 152190 nM T53585 CIL0S7 46906558 IC50 = 750 nM T53585 C15CDK 53231152 IC50 = 24.55 nM T53585 CDHF72 67869066 IC50 = 20 nM T53585 C4MH6F 67869344 IC50 = 7.5 nM T53585 CSKE34 67869518 IC50 = 10 nM T53585 CJN9B6 71461154 IC50 = 22300 nM T53585 CU65GH 71655059 IC50 = 54.1 nM T53585 CPS58L 71655136 IC50 = 16.8 nM T53585 CFW7Q9 71655137 IC50 = 13.1 nM T53585 C9S0UB 71655138 IC50 = 12.3 nM T53585 CU27EV 71655139 IC50 = 43.7 nM T53585 CO8R1Z 71655216 IC50 = 36.5 nM T53585 C0W6EK 71655283 IC50 = 53.8 nM T53585 C67TKL 73345785 IC50 = 0.83 nM T53585 C87BDJ 73346768 IC50 = 17 nM T53585 CRX43H 73347269 IC50 = 0.106 nM T53585 CUYA31 73348279 IC50 = 62 nM T53585 C7WVI9 73352866 IC50 = 26 nM T53585 CG1CA0 73352867 IC50 = 50 nM T53585 C3AH7Q 73354373 IC50 = 18 nM T53585 C7B6XC 73355938 IC50 = 150 nM T53585 CWT42G 118708583 IC50 = 8.892 nM T53585 C12TWI 118717838 IC50 = 44.67 nM T53585 CS0WH1 118718594 IC50 = 13.3 nM T53585 CAOS68 118718595 IC50 = 19.7 nM T53585 CQK5M3 118718596 IC50 = 7.6 nM T53585 C7IS4F 118718597 IC50 = 10.8 nM T53585 C5TZH7 132521485 IC50 = 387000 nM T53585 D00RHH 24916963 IC50 = 0.3 nM T53585 D00TIO 44331923 IC50 = 1.8 nM T53585 D00UOI 56947030 IC50 = 0.2 nM T53585 D01WQF 46906163 IC50 = 1470 nM T53585 D01YQX 14309408 IC50 = 7000 nM T53585 D01ZAL 44370459 IC50 = 370 nM T53585 D02MEX 56947026 IC50 = 0.57 nM T53585 D03CYY 24873518 IC50 = 1520 nM T53585 D03EAN 56947035 IC50 = 0.05 nM T53585 D05GWF 56947027 IC50 = 0.27 nM T53585 D05UQC 73348335 IC50 = 4.8 nM T53585 D05YUT 44354270 IC50 = 1000 nM T53585 D06FRE 56947041 IC50 = 3500 nM T53585 D06OVX 65094 IC50 = 300 nM T53585 D07QAX 14849849 IC50 = 5.7 nM T53585 D08SKU 14309407 IC50 = 5000 nM T53585 D09CSQ 46906168 Ki = 51 nM T53585 D09EBV 14309406 IC50 = 3000 nM T53585 D09QIA 68167 IC50 = 5000 nM T53585 D0A6FX 14309404 IC50 = 2000 nM T53585 D0B2FM 25254901 IC50 = 19430 nM T53585 D0C1RY 24873519 IC50 = 1780 nM T53585 D0C5LO 5312662 IC50 = 5000 nM T53585 D0C8HK 9543636 IC50 = 500 nM T53585 D0CU3I 14309405 IC50 = 3000 nM T53585 D0G4ZG 56947023 IC50 = 0.018 nM T53585 D0G6PS 56947029 IC50 = 1.9 nM T53585 D0IJ7H 1662 Ki = 23.5 nM T53585 D0M9BZ 56947040 IC50 = 250 nM T53585 D0NU6K 9543637 IC50 = 1500 nM T53585 D0O2FD 56947039 IC50 = 30 nM T53585 D0Q6WP 44392476 IC50 = 8.7 nM T53585 D0S1LA 25254902 IC50 = 16940 nM T53585 D0T4PL 56947038 IC50 = 0.5 nM T53585 D0W5FM 15931922 IC50 = 1400 nM T53585 D0X0GV 44452237 IC50 = 22310 nM T53585 D0X1VL 44452269 IC50 = 3840 nM T58937 D05WWJ 6604909 IC50 = 1800 nM T58937 D0O0BM 44156901 IC50 > 10000 nM T58937 C16UJV 2916853 EC50 = 11400 nM T58937 C7B2UD 4154232 IC50 = 518 nM T58937 CL5BU6 4639181 IC50 = 478 nM T58937 C4PJ1X 5311286 IC50 = 214 nM T58937 CUY2A3 5311287 IC50 = 3.8 nM T58937 C3TR2C 6436908 IC50 = 500 nM T58937 CK1OS6 6437024 IC50 = 29.2 nM T58937 CCH5V1 6913738 IC50 = 4350 nM T58937 C9LY7V 8194613 IC50 > 10000 nM T58937 C8Z6VJ 9225008 EC50 = 14200 nM T58937 CX82ZB 9502378 IC50 = 2816 nM T58937 CH0O9S 10024067 IC50 = 170 nM T58937 CFT5R0 10048123 IC50 = 30 nM T58937 CW46IX 10476003 IC50 = 33 nM T58937 CAY47E 10882694 IC50 = 696 nM T58937 CZS7V2 10915847 IC50 = 77 nM T58937 CA09SY 11014349 IC50 = 2313 nM T58937 C7CW0X 11046680 IC50 = 2563 nM T58937 CJC0X3 11058466 IC50 = 566 nM T58937 C7JP0L 11058608 IC50 = 1321 nM T58937 CKL5O9 11059011 IC50 = 84 nM T58937 C76YFB 11155030 EC50 > 30000 nM T58937 CFO4R6 11155673 IC50 > 30000 nM T58937 CH72UP 11156047 EC50 > 30000 nM T58937 CUBX19 11189444 EC50 > 30000 nM T58937 CS5ET8 11212373 EC50 > 30000 nM T58937 C26MVG 11223982 EC50 > 30000 nM T58937 C2EY1P 11237095 EC50 > 30000 nM T58937 CX43IH 11248146 EC50 > 30000 nM T58937 CQR3W4 11283425 EC50 = 24000 nM T58937 C8S4FU 11317045 EC50 > 30000 nM T58937 CS1W7V 11338717 EC50 > 30000 nM T58937 CQC4G5 11372671 EC50 > 30000 nM T58937 CV71EO 11396919 EC50 = 4800 nM T58937 C3NWX6 11405950 IC50 > 30000 nM T58937 CGO58L 11406629 EC50 = 7000 nM T58937 CBJ0X5 11407510 EC50 > 30000 nM T58937 CW0E4L 11418847 EC50 > 30000 nM T58937 CKIQ83 11463791 EC50 > 30000 nM T58937 CC9TX5 11464294 EC50 > 30000 nM T58937 CP0AY1 11465204 EC50 = 4000 nM T58937 CRU3C9 11465585 EC50 > 30000 nM T58937 CAY3P0 11488045 EC50 > 30000 nM T58937 C9N7BP 11488921 EC50 > 30000 nM T58937 CYFU19 11496738 IC50 > 30000 nM T58937 CHV9P4 11503316 IC50 > 30000 nM T58937 CWNS78 11503732 IC50 > 30000 nM T58937 C8K6LT 11503999 IC50 > 30000 nM T58937 CGWZ71 11510618 IC50 > 30000 nM T58937 C0P9VC 11517722 IC50 > 30000 nM T58937 CMEK74 11518581 EC50 > 30000 nM T58937 C4OAQ8 11518805 EC50 > 30000 nM T58937 CHGW75 11539784 IC50 > 30000 nM T58937 CW2IZ4 11540267 EC50 > 30000 nM T58937 C2JQ1P 11569401 EC50 = 12000 nM T58937 C9CT2I 11583046 IC50 > 30000 nM T58937 CAR70B 11583581 IC50 > 30000 nM T58937 CELV43 11597407 EC50 > 30000 nM T58937 C4NMD3 11619325 IC50 > 30000 nM T58937 C41ASM 11620014 IC50 > 30000 nM T58937 C6SPR0 11627103 EC50 > 30000 nM T58937 CIJ40B 11641798 EC50 > 30000 nM T58937 CJ6PI1 11647944 EC50 > 30000 nM T58937 C8R4DN 11656017 IC50 > 10000 nM T58937 CHBN05 11662843 IC50 > 30000 nM T58937 CKI68D 11663033 EC50 > 30000 nM T58937 CW9H0I 11677151 IC50 > 30000 nM T58937 C01ORH 11691531 EC50 > 30000 nM T58937 CWK01R 11699068 IC50 > 30000 nM T58937 CYW07F 11732786 IC50 = 1563 nM T58937 CV8CF3 11749578 EC50 = 25000 nM T58937 C3IF8B 11953816 IC50 = 600 nM T58937 C4I3RS 12307852 IC50 = 33200 nM T58937 CD7K0Y 15965865 EC50 = 12000 nM T58937 C4YMP1 16725956 IC50 = 319 nM T58937 C2L9HN 16960944 EC50 = 24500 nM T58937 C9EAP4 18098131 EC50 = 2000 nM T58937 C87WIK 18104758 EC50 = 27000 nM T58937 C8AZW7 18441735 EC50 = 72000 nM T58937 COSK18 23544093 IC50 = 320 nM T58937 CK7F6P 23544094 IC50 = 130 nM T58937 CO6VK5 23544101 IC50 = 1200 nM T58937 C34WTK 23544106 IC50 = 330 nM T58937 CH31CE 23544108 IC50 = 4000 nM T58937 CIG6H8 23544109 IC50 = 3400 nM T58937 CLY24K 23544123 IC50 = 1600 nM T58937 CS7DZ3 23544124 IC50 = 130 nM T58937 C2GZQ5 23544125 IC50 = 370 nM T58937 CSQ95N 23544126 IC50 = 140 nM T58937 CFJK60 23544127 IC50 = 56 nM T58937 CDZ9T2 23544128 IC50 = 140 nM T58937 C75WGA 23544131 IC50 = 86 nM T58937 CZN23Y 23544133 IC50 = 1600 nM T58937 C1JAF3 23544135 IC50 = 1200 nM T58937 CGS67N 23544168 IC50 = 670 nM T58937 C2CDW3 23544173 IC50 = 1100 nM T58937 C0OCU2 23544175 IC50 = 1800 nM T58937 C9LR3W 23544177 IC50 = 4400 nM T58937 C85DUO 23544186 IC50 = 130 nM T58937 CEGQ70 23544187 IC50 = 43 nM T58937 C9AJB2 23544188 IC50 = 81 nM T58937 CXP6C5 23544189 IC50 = 1400 nM T58937 C2JC5L 23544201 IC50 = 24 nM T58937 C8UEB5 23544202 IC50 = 89 nM T58937 C39TCP 23544204 IC50 = 67 nM T58937 CT9E7R 23544205 IC50 = 3400 nM T58937 C37TYI 23544211 IC50 = 58 nM T58937 CB01MP 23544212 IC50 = 1900 nM T58937 CTFO41 23544287 IC50 = 120 nM T58937 CR0W4K 23544296 IC50 = 99 nM T58937 CCDV64 23544305 IC50 = 77 nM T58937 CFP0K9 23544311 IC50 = 2400 nM T58937 C3JIY0 23544313 IC50 = 4100 nM T58937 CS7E2L 24532923 EC50 = 1400 nM T58937 CZ03FI 24649020 EC50 = 11400 nM T58937 CQ35ZB 24743795 EC50 = 6650 nM T58937 CYM02E 24847114 EC50 > 30000 nM T58937 CDI7N3 24897002 EC50 = 14100 nM T58937 C8GN9W 24899993 EC50 = 14800 nM T58937 CIZ6O1 24900235 EC50 = 7520 nM T58937 C61ARF 24900236 EC50 = 9570 nM T58937 C7UD6F 24957934 IC50 > 30000 nM T58937 C8U4KM 26365758 EC50 = 3100 nM T58937 CR8IG7 29297108 EC50 = 300 nM T58937 CTEN36 40846579 IC50 = 9000 nM T58937 CO74NY 41772744 EC50 > 30000 nM T58937 CPF50A 44184875 EC50 > 30000 nM T58937 C8ARJ4 44190514 IC50 = 496 nM T58937 C0GKY6 44367213 IC50 > 10000 nM T58937 CC7M9G 44367338 IC50 ~ 10000 nM T58937 CY2R0F 44367350 IC50 > 5000 nM T58937 CLU91D 44367423 IC50 > 5000 nM T58937 C01XQP 44367437 IC50 = 300 nM T58937 C08LCI 44367547 IC50 > 5000 nM T58937 C53YJA 44367548 IC50 > 5000 nM T58937 CYPU73 44367563 IC50 > 10000 nM T58937 CG7A9P 44367564 IC50 > 5000 nM T58937 CW9QG2 44406457 EC50 = 25000 nM T58937 CGN73V 44406458 EC50 > 100000 nM T58937 C0J7IK 44406489 EC50 = 12000 nM T58937 C5TIM4 44406497 EC50 = 16000 nM T58937 CBUR32 44406503 EC50 = 36000 nM T58937 C17FYG 44406538 EC50 = 72000 nM T58937 C07CNE 44406539 EC50 = 67000 nM T58937 C5DGV2 44406540 EC50 = 21000 nM T58937 C9Z0ET 44406541 EC50 = 2500 nM T58937 C1L8CG 44406543 EC50 = 19000 nM T58937 CP1OZ6 44406544 EC50 = 25000 nM T58937 CR5WZ2 44406546 EC50 > 100000 nM T58937 CS04TK 44406550 EC50 = 41000 nM T58937 C8HRC9 44406551 EC50 > 100000 nM T58937 C8XHL1 44406552 EC50 = 3400 nM T58937 C21FWX 44406553 EC50 = 27000 nM T58937 C1LVU2 44406558 EC50 > 100000 nM T58937 CPG5O7 44406559 EC50 = 9000 nM T58937 CEI1H6 44406577 EC50 > 100000 nM T58937 CD7Y0Z 44406585 EC50 = 35000 nM T58937 CC15BY 44406587 EC50 = 6000 nM T58937 C2MV0K 44406589 EC50 = 24000 nM T58937 C1IM9R 44406603 EC50 = 57000 nM T58937 C3VE8N 44406604 EC50 = 70000 nM T58937 C2JG5K 44406608 EC50 = 15000 nM T58937 CCI5Z1 44406618 EC50 = 10000 nM T58937 C7ES2W 44406621 EC50 = 26000 nM T58937 C0MX1J 44406626 EC50 > 100000 nM T58937 C0SKT9 44406641 EC50 = 18000 nM T58937 CHF65L 44406659 EC50 = 13000 nM T58937 CZNQ19 44406672 EC50 = 23000 nM T58937 C38ABN 44406682 EC50 = 35000 nM T58937 CZ65PF 44406685 EC50 > 100000 nM T58937 COHV70 44406692 EC50 = 11000 nM T58937 CMR3C6 44406693 EC50 = 25000 nM T58937 CIR94D 44406707 EC50 = 16000 nM T58937 CC1A9V 44406708 EC50 = 5000 nM T58937 CB36AF 44406709 EC50 = 15000 nM T58937 C4M1GV 44406714 EC50 = 24000 nM T58937 CWY76P 44406719 EC50 = 2900 nM T58937 CC6SW1 44406725 EC50 = 2600 nM T58937 CYA4I3 44406726 EC50 = 6800 nM T58937 C6O2VL 44414730 EC50 = 39630 nM T58937 CRCQ06 44414830 EC50 > 30000 nM T58937 C1PK7O 44414844 EC50 = 8360 nM T58937 C5Z9VE 44414845 EC50 = 39950 nM T58937 C4LI9Q 44414865 EC50 = 16680 nM T58937 CDEC-35 44420018 IC50 > 30000 nM T58937 CLJ58G 44420020 IC50 > 30000 nM T58937 CJP9Y2 44420021 IC50 > 30000 nM T58937 CZ54MW 44420030 IC50 > 30000 nM T58937 C69SHV 44420039 IC50 > 30000 nM T58937 CVL2E6 44420041 IC50 > 30000 nM T58937 CQ43MW 44420042 IC50 > 30000 nM T58937 C2ETD8 44420043 IC50 > 30000 nM T58937 C65CVW 44420046 IC50 > 30000 nM T58937 C5K7BH 44420047 IC50 > 30000 nM T58937 CE20MW 44420048 IC50 > 30000 nM T58937 CLWG78 44420049 IC50 > 30000 nM T58937 CCB3V7 44420052 IC50 > 30000 nM T58937 CW90RA 44420055 IC50 > 30000 nM T58937 CWKV41 44420132 IC50 > 30000 nM T58937 C8AZ0R 44420133 IC50 > 30000 nM T58937 C8ILS1 44420139 IC50 > 30000 nM T58937 C7H0UM 44420140 IC50 > 30000 nM T58937 CP2YG8 44423663 IC50 = 1230 nM T58937 CUB30F 44438465 IC50 = 531 nM T58937 CE36YV 44438467 IC50 = 31.5 nM T58937 CI93VE 44438472 IC50 = 385 nM T58937 CXD9B1 44438473 IC50 = 401 nM T58937 C0QEB9 44438474 IC50 = 857 nM T58937 C8MJX3 44444240 IC50 > 30000 nM T58937 CY1M5B 44444241 IC50 > 30000 nM T58937 CJ4MN5 44444243 IC50 > 30000 nM T58937 C2PD4R 44444244 IC50 > 30000 nM T58937 C1DG6B 44444245 IC50 > 30000 nM T58937 CP20CO 44444246 IC50 > 30000 nM T58937 CSK28U 44444247 IC50 > 30000 nM T58937 C3QTF8 44444248 IC50 > 30000 nM T58937 CM08FN 44444249 IC50 > 30000 nM T58937 C39BVE 44444250 IC50 > 30000 nM T58937 CA1YH0 44444251 IC50 > 30000 nM T58937 C6EQ9M 44444254 IC50 > 30000 nM T58937 CB6Q4T 44444255 IC50 > 30000 nM T58937 CXEP90 44444258 IC50 > 30000 nM T58937 CUI25H 44444260 IC50 > 30000 nM T58937 C0R3PZ 44444261 IC50 > 30000 nM T58937 C1W5TQ 44444262 IC50 > 30000 nM T58937 CT9O7J 44444263 IC50 > 30000 nM T58937 C1QIO5 44444264 IC50 > 30000 nM T58937 C9NDY4 44444265 IC50 > 30000 nM T58937 CRI72W 44444267 IC50 > 30000 nM T58937 CS9R1C 44444268 IC50 > 30000 nM T58937 CUF89R 44444270 IC50 > 30000 nM T58937 CA1O3V 44444271 IC50 > 30000 nM T58937 CJSA47 44444273 IC50 > 30000 nM T58937 CHUJ64 44444275 IC50 > 30000 nM T58937 CCMV69 44444276 IC50 > 30000 nM T58937 C4X3EO 44444281 IC50 > 30000 nM T58937 CX46JK 44444284 IC50 > 30000 nM T58937 C7QHD4 44444287 IC50 > 30000 nM T58937 C29RVP 44444289 IC50 > 30000 nM T58937 CI0D3P 44444290 IC50 > 30000 nM T58937 CI1T0P 44444291 IC50 > 30000 nM T58937 C3Y5MT 44444292 IC50 > 30000 nM T58937 CUAK74 44444294 IC50 > 30000 nM T58937 CX47CG 44444296 IC50 > 30000 nM T58937 C2GF7J 44444298 IC50 > 30000 nM T58937 CA87MB 44564635 IC50 > 30000 nM T58937 CDC0B2 44564672 IC50 > 30000 nM T58937 CF2TP7 44564679 IC50 > 30000 nM T58937 CTJ49O 44564680 IC50 > 30000 nM T58937 CCL8B7 44564681 IC50 > 30000 nM T58937 CQN60Y 44564766 IC50 > 30000 nM T58937 C5VIN0 44565248 IC50 > 30000 nM T58937 COR7F4 44565249 IC50 > 30000 nM T58937 CS2I4V 44565250 IC50 > 30000 nM T58937 C7FE5L 44565251 IC50 > 30000 nM T58937 C20DZB 44565252 IC50 > 30000 nM T58937 C7URY2 44565253 IC50 > 30000 nM T58937 CQV4K2 44565260 IC50 > 30000 nM T58937 CG21WE 44565261 IC50 > 30000 nM T58937 C4PAC2 44565262 IC50 > 30000 nM T58937 C2XJY7 44565263 IC50 > 30000 nM T58937 CH4GW0 44565264 IC50 > 30000 nM T58937 C8I3SF 44565265 IC50 > 30000 nM T58937 C7WL4C 44565270 IC50 > 30000 nM T58937 CC1O6M 44565271 IC50 > 30000 nM T58937 C6EAC3 44565272 IC50 > 30000 nM T58937 CG80OC 44578914 EC50 = 29200 nM T58937 CBG04P 44578955 EC50 = 4200 nM T58937 CA3FO8 44578956 EC50 = 19100 nM T58937 CA16QJ 44578957 EC50 = 23100 nM T58937 C4KI0B 44579189 EC50 > 30000 nM T58937 C1O5ET 44579232 EC50 > 30000 nM T58937 CO7MU4 44580053 EC50 > 30000 nM T58937 CY7MA0 44580054 EC50 = 13400 nM T58937 CI24ZU 44580055 EC50 = 11200 nM T58937 C86GWQ 44580106 EC50 > 30000 nM T58937 CF5ST4 44580229 EC50 = 8300 nM T58937 CH1G5K 44580230 EC50 = 4000 nM T58937 CBLJ49 44580260 EC50 = 7700 nM T58937 C1UO6X 44580261 EC50 = 1170 nM T58937 C1FNB8 44580262 EC50 = 3300 nM T58937 CYA4U0 44580302 EC50 = 1100 nM T58937 C4EK3O 44580303 EC50 = 2100 nM T58937 COY93Q 44580304 EC50 = 4300 nM T58937 CX16RS 44580305 EC50 > 30000 nM T58937 CD9M8A 44580340 EC50 = 29000 nM T58937 CT5FH1 44580341 EC50 = 15000 nM T58937 CBJ63S 44580511 EC50 > 30000 nM T58937 C1NME3 44580512 EC50 > 30000 nM T58937 CRCG05 44580513 EC50 = 5100 nM T58937 CLT4V2 44580551 EC50 = 11000 nM T58937 CA92XB 44580552 EC50 = 13000 nM T58937 CZK47O 44580553 EC50 > 30000 nM T58937 C8YI9V 44580554 EC50 > 30000 nM T58937 C54RAU 44580597 EC50 > 30000 nM T58937 CAU6P2 44580598 EC50 > 30000 nM T58937 C0PFY1 44580672 EC50 = 3300 nM T58937 C1Z8FK 44580673 EC50 = 10000 nM T58937 C9KY5O 44580713 EC50 = 8500 nM T58937 CB1HZ6 44580752 EC50 > 30000 nM T58937 C7L8JD 44580753 EC50 > 30000 nM T58937 CB7FS6 44580754 EC50 > 30000 nM T58937 C18RQM 44591636 IC50 > 10000 nM T58937 CMTH41 44591637 IC50 > 10000 nM T58937 CY47VM 44591699 IC50 > 10000 nM T58937 C91NGO 44591734 IC50 > 10000 nM T58937 C05LWQ 44591764 IC50 > 10000 nM T58937 CCA7K5 44593648 EC50 = 5900 nM T58937 C14LUA 45267039 IC50 > 10000 nM T58937 CU0JM3 45267807 IC50 > 10000 nM T58937 CUEY48 45267808 IC50 > 10000 nM T58937 C18EGU 45268687 IC50 > 10000 nM T58937 CS67XW 45270376 IC50 > 10000 nM T58937 CU4OH2 45270377 IC50 > 10000 nM T58937 CH17KU 45272913 IC50 = 1150 nM T58937 CPUR70 45272936 IC50 > 10000 nM T58937 CQ98IX 45272939 IC50 > 10000 nM T58937 C9FS6T 46213935 IC50 > 30000 nM T58937 CL51NF 46216732 IC50 = 6250 nM T58937 CZJL95 46216733 IC50 > 10000 nM T58937 C1DO4U 46230960 IC50 = 4200 nM T58937 C59XOB 46230961 IC50 = 1170 nM T58937 C9EGU1 46230962 IC50 = 2270 nM T58937 C7G3TB 46231012 IC50 = 2210 nM T58937 C1J0WY 46231013 IC50 > 10000 nM T58937 C2FVA8 46231075 IC50 > 3450 nM T58937 CA3R5W 46231076 IC50 > 7290 nM T58937 CSZ2F6 46231077 IC50 = 3000 nM T58937 CVL6C0 46231146 IC50 > 10000 nM T58937 C8W4VL 46231147 IC50 = 3020 nM T58937 CRTO63 46231148 IC50 = 3880 nM T58937 CZ6C0S 46231149 IC50 = 8870 nM T58937 CTQ38S 46239398 IC50 > 30000 nM T58937 C93GVI 46239399 IC50 > 30000 nM T58937 CY7S3X 46239400 IC50 > 30000 nM T58937 C4ER1X 46239401 IC50 > 30000 nM T58937 CX04CO 46239402 IC50 > 30000 nM T58937 CT14BG 46239503 IC50 > 30000 nM T58937 CK93AJ 46239504 IC50 > 30000 nM T58937 COV4I9 46239505 IC50 > 30000 nM T58937 CO9YC0 46239506 IC50 > 30000 nM T58937 C04GRB 46239507 IC50 > 30000 nM T58937 C1NG0Y 46239508 IC50 > 30000 nM T58937 CC98ZF 46837246 EC50 > 30000 nM T58937 C0GY1V 46837247 EC50 > 30000 nM T58937 CQ41PO 46837248 EC50 > 30000 nM T58937 CN1EK8 46837249 EC50 > 30000 nM T58937 C5UL9K 46837250 EC50 > 30000 nM T58937 CB01AC 46837364 EC50 = 29000 nM T58937 C6IXU7 46837365 EC50 > 30000 nM T58937 CRF5X4 46838883 EC50 > 30000 nM T58937 CVS8X0 46838884 EC50 > 30000 nM T58937 C8FZ1X 46838885 EC50 > 30000 nM T58937 C6ACV2 46838886 EC50 > 30000 nM T58937 CK06VF 46839028 EC50 > 30000 nM T58937 C0M8AW 46839029 EC50 > 30000 nM T58937 C1ZDW9 46839030 EC50 > 30000 nM T58937 CZ85PM 46839031 EC50 > 30000 nM T58937 C4PE5H 46839032 EC50 > 30000 nM T58937 C3L0MZ 46839160 EC50 > 30000 nM T58937 C6K7FV 46839161 EC50 > 30000 nM T58937 CT51HS 46839162 EC50 > 30000 nM T58937 CPI82F 46839163 EC50 > 30000 nM T58937 C21ILB 46839164 EC50 > 30000 nM T58937 C1OIG5 46839165 EC50 > 30000 nM T58937 CB93RG 46839296 EC50 > 30000 nM T58937 CS09WQ 46839297 EC50 > 30000 nM T58937 C9S4IH 46839298 EC50 > 30000 nM T58937 CA0MR4 46839299 EC50 > 30000 nM T58937 C1EPB3 46839300 EC50 = 24200 nM T58937 C2UYK7 46850264 EC50 = 15000 nM T58937 CP7HF9 46907933 IC50 = 340 nM T58937 CUL54V 46912220 IC50 > 30000 nM T58937 C40LTM 46912222 IC50 > 30000 nM T58937 C3AF9Y 46917638 IC50 = 1170 nM T58937 C2DO4V 46935693 IC50 > 30000 nM T58937 C4DJ1R 46935694 IC50 > 30000 nM T58937 CIN62E 46935749 IC50 > 30000 nM T58937 CP9JK2 46938091 IC50 > 30000 nM T58937 C5G6IO 46938092 IC50 > 30000 nM T58937 CLC63O 46938152 IC50 > 30000 nM T58937 C5I1HQ 49798777 EC50 > 30000 nM T58937 CR9N2O 52922059 IC50 = 214 nM T58937 CF7KW0 52922061 IC50 = 54.6 nM T58937 CLB47C 52922067 IC50 = 143 nM T58937 CUY3G2 52922080 IC50 = 613 nM T58937 CO4AW2 53317349 EC50 > 30000 nM T58937 CB4J9Y 53317462 EC50 > 30000 nM T58937 C2NQJ0 53318186 EC50 > 30000 nM T58937 C5VTR7 53318583 EC50 > 30000 nM T58937 CXY8A4 53319905 EC50 = 30000 nM T58937 C65DNJ 53319906 EC50 > 30000 nM T58937 C7PL6F 53319952 EC50 > 30000 nM T58937 C0W2AF 53321255 EC50 > 30000 nM T58937 CO6N5I 53321256 EC50 > 30000 nM T58937 C6HIS7 53322576 EC50 > 30000 nM T58937 CA24UX 53323869 EC50 = 14300 nM T58937 CDU0B3 53323870 EC50 > 30000 nM T58937 CAM5B9 53323918 EC50 > 30000 nM T58937 C89NPM 53325153 EC50 > 30000 nM T58937 CI3GU2 53325154 EC50 > 30000 nM T58937 C6Y4PN 53325155 EC50 > 30000 nM T58937 C40KDP 53326450 EC50 > 30000 nM T58937 C0GT4H 53326451 EC50 > 30000 nM T58937 C89ZWP 54764172 IC50 > 75000 nM T58937 CDJ48K 54764173 IC50 > 75000 nM T58937 CNC14G 54764522 IC50 > 75000 nM T58937 CF0NC5 54764945 IC50 > 75000 nM T58937 CN62OP 54764946 IC50 > 75000 nM T58937 CH57OM 54765031 IC50 > 75000 nM T58937 C9J7AT 56658396 IC50 = 10000 nM T58937 CIW3R2 56658557 IC50 > 25118.86 nM T58937 CZU30J 56658558 IC50 = 12589.25 nM T58937 C2XRE3 56658559 IC50 > 25118.86 nM T58937 CNY8K3 56658560 IC50 = 19952.62 nM T58937 CH73OR 56658561 IC50 > 25118.86 nM T58937 CTKI43 56658562 IC50 > 25118.86 nM T58937 CXH0V2 56661885 IC50 > 25118.86 nM T58937 C1ZNL5 56662010 IC50 > 25118.86 nM T58937 C6OHX7 56662011 IC50 > 25118.86 nM T58937 C89FMR 56662012 IC50 = 7943.28 nM T58937 CYJ23N 56662013 IC50 = 19952.62 nM T58937 C15LNY 56662014 IC50 > 25118.86 nM T58937 C9QE1S 56665356 IC50 > 25118.86 nM T58937 C08ALR 56665500 IC50 > 25118.86 nM T58937 CD7PK4 56665501 IC50 > 25118.86 nM T58937 CT5I3H 56665502 IC50 = 15848.93 nM T58937 C07VIA 56665503 IC50 > 6309.57 nM T58937 COR3T2 56668927 IC50 > 25118.86 nM T58937 CDM63Q 56668928 IC50 = 15848.93 nM T58937 C6QRE1 56668929 IC50 > 25118.86 nM T58937 CA5UB3 56672410 IC50 > 25118.86 nM T58937 C6W2PY 56672411 IC50 > 25118.86 nM T58937 CU49AH 56672412 IC50 = 5011.87 nM T58937 CV6FC0 56675655 IC50 > 25118.86 nM T58937 C1GFE0 56679109 IC50 > 19952.62 nM T58937 CGD58R 56679110 IC50 > 25118.86 nM T58937 CQXO18 57557335 IC50 = 3800 nM T58937 CG1MS3 70685518 EC50 > 30000 nM T58937 CY6E2Q 70691339 EC50 = 25000 nM T58937 C9EIY7 71566778 IC50 = 860 nM T58937 CMET87 71584823 IC50 = 105 nM T58937 CUX5O9 71585152 IC50 = 79.6 nM T58937 CWL2G6 71585155 IC50 = 15.3 nM T58937 C0EF5K 71585157 IC50 = 62.1 nM T58937 CVQZ85 71716253 IC50 > 75000 nM T58937 CUP19I 71716254 IC50 > 75000 nM T58937 CZHI20 71718079 IC50 > 75000 nM T58937 CV2Z7K 71718685 IC50 > 75000 nM T58937 C97SYX 71718694 IC50 > 75000 nM T58937 CKC70J 71719305 IC50 > 75000 nM T58937 C72ADI 71719306 IC50 > 75000 nM T58937 CV68AD 71719905 IC50 > 75000 nM T58937 C3JAD2 71720525 IC50 > 75000 nM T58937 COVM31 71720526 IC50 > 75000 nM T58937 CND02X 76310572 IC50 > 30000 nM T58937 CD20WP 76310588 IC50 > 30000 nM T58937 C6NST3 76314240 IC50 > 30000 nM T58937 C5YML9 76314241 IC50 > 30000 nM T58937 C6KU8P 76317794 IC50 > 30000 nM T58937 CG8H0J 76317812 IC50 > 30000 nM T58937 CIO7F4 76321506 IC50 > 30000 nM T58937 CJTX79 76321522 IC50 > 30000 nM T58937 CN1E8K 76321523 IC50 > 30000 nM T58937 C7R2YC 76325123 IC50 > 30000 nM T58937 CNIT93 76325124 IC50 > 30000 nM T58937 CV18IA 76328662 IC50 > 30000 nM T58937 C36ULS 76328663 IC50 > 30000 nM T58937 C1WEM6 76328673 IC50 > 30000 nM T58937 CZ5I8G 76328674 IC50 > 30000 nM T58937 CM23TB 76332339 IC50 > 30000 nM T58937 C6U2PQ 76335977 IC50 > 30000 nM T58937 CJ57DZ 86745788 IC50 = 64.8 nM T58937 CZK18W 88463909 IC50 = 865 nM T58937 C2T4XJ 88494111 IC50 = 2330 nM T58937 C01UNB 90665166 IC50 = 1150 nM T58937 C5FTW2 99116834 IC50 = 259 nM T58937 C9ME7U 117897388 IC50 > 75000 nM T58937 C38JEB 117897542 IC50 > 75000 nM T58937 C3PUR8 117897549 IC50 > 75000 nM T58937 C89EQN 117897570 IC50 > 75000 nM T58937 CSXH08 117897680 IC50 > 75000 nM T58937 C2ED0W 117897772 IC50 > 75000 nM T58937 C5N2SK 117897780 IC50 > 75000 nM T58937 C4A6JK 117897787 IC50 > 75000 nM T58937 CVK03J 117897796 IC50 > 75000 nM T58937 C30EKF 117897864 IC50 > 75000 nM T58937 CIT13E 117897929 IC50 > 75000 nM T58937 CU2V9L 117897938 IC50 > 75000 nM T58937 C4CH1E 117897955 IC50 > 75000 nM T58937 CA1Z6P 117897961 IC50 > 75000 nM T58937 CJ42DF 117897992 IC50 > 75000 nM T58937 CMI40T 117898061 IC50 > 75000 nM T58937 CV47YD 117898069 IC50 > 75000 nM T58937 CGY40U 117898099 IC50 > 75000 nM T58937 CA2L7N 117898102 IC50 > 75000 nM T58937 CL3PM6 117898113 IC50 > 75000 nM T58937 C7DLZ6 117898161 IC50 > 75000 nM T58937 CO0K9G 117898177 IC50 > 75000 nM T58937 C2U0FV 117898180 IC50 > 75000 nM T58937 CAEK03 117898196 IC50 > 75000 nM T58937 C2T9EV 117898210 IC50 > 75000 nM T58937 CRV8S3 118478927 IC50 > 10000 nM T58937 CL32JE 118478933 IC50 > 10000 nM T58937 C5S1HZ 118478972 IC50 > 10000 nM T58937 C8G9HP 118478986 IC50 > 10000 nM T58937 CBV89G 118478994 IC50 > 10000 nM T58937 CK0ER5 118478999 IC50 > 10000 nM T58937 CU25KC 118479000 IC50 > 10000 nM T58937 CW07IS 118479006 IC50 > 10000 nM T58937 C3ZAV0 118479034 IC50 > 10000 nM T58937 C4W6ZS 118479038 IC50 > 10000 nM T58937 CRG24C 118479053 IC50 > 10000 nM T58937 CD4ME1 118479123 IC50 > 10000 nM T58937 CB0XM2 118479161 IC50 > 10000 nM T58937 C18NTQ 118479199 IC50 > 10000 nM T58937 CJ0Z1Y 118479222 IC50 > 10000 nM T58937 CP0U6Y 118479229 IC50 > 10000 nM T58937 C3A6HD 118479231 IC50 > 10000 nM T58937 CJ14CR 118479241 IC50 > 10000 nM T58937 C1FO3N 118479293 IC50 > 10000 nM T58937 CF02TZ 118479295 IC50 > 10000 nM T58937 C90TED 118479305 IC50 > 10000 nM T58937 C7I9RC 118479316 IC50 > 10000 nM T58937 CRC4F6 118479354 IC50 > 10000 nM T58937 CRCV51 118479359 IC50 > 10000 nM T58937 CJL5W0 118479428 IC50 > 10000 nM T58937 CS2VA7 118479440 IC50 > 10000 nM T58937 CJ9P0M 118479445 IC50 > 10000 nM T58937 C3U1RB 118479452 IC50 > 10000 nM T58937 C1O2IB 118710993 IC50 = 4040 nM T58937 CV3UX0 118710994 IC50 = 516 nM T58937 CK8CG6 118710995 IC50 = 250 nM T58937 CJ94ED 118710996 IC50 = 2200 nM T58937 C3WV7H 118710997 IC50 = 2800 nM T58937 CBR96I 118710998 IC50 = 879 nM T58937 CF40CB 118710999 IC50 = 2320 nM T58937 CRYG59 118711000 IC50 = 440 nM T58937 CA45CF 118711001 IC50 = 112 nM T58937 CL9F4G 118711002 IC50 = 431 nM T58937 CHI54T 118711003 IC50 = 869 nM T58937 C92RQA 118711004 IC50 = 361 nM T58937 CYDZ23 118711005 IC50 = 115 nM T58937 CIWS86 118711006 IC50 = 363 nM T58937 CD0O5X 118711007 IC50 = 71.4 nM T58937 C5XWV2 118711008 IC50 = 330 nM T58937 CK2S3B 118711009 IC50 = 107 nM T58937 CR86ZJ 118711010 IC50 = 99.1 nM T58937 CHZ6X5 118711011 IC50 = 65.8 nM T58937 CU0JO9 118711012 IC50 = 181 nM T58937 C90MNZ 118711013 IC50 = 51.9 nM T58937 CT9K0V 124000588 IC50 > 10000 nM T58937 COA0U2 135239967 IC50 = 1000 nM T58937 CE10YC 135239972 IC50 > 10000 nM T58937 CGEV09 135239984 IC50 = 259 nM T58937 CY14GZ 135239991 IC50 = 151 nM T58937 C91VJQ 135239995 IC50 > 10000 nM T58937 CL0S6Q 135240007 IC50 = 1810 nM T58937 C4E7OH 135240008 IC50 = 3750 nM T58937 C13CQX 135240011 IC50 > 30000 nM T58937 C6OI3K 145973962 IC50 > 10000 nM T58937 CBC0F5 154026493 IC50 > 10000 nM T58937 C16LXF 155521483 IC50 > 75000 nM T58937 C10YRG 155524872 IC50 > 75000 nM T58937 C4WJ0I 155525087 IC50 > 75000 nM T58937 C8AU6P 155542971 IC50 > 75000 nM T58937 C93OTJ 155546926 IC50 > 75000 nM T58937 CZT3W7 155547990 IC50 = 48.3 nM T58937 C7NLE5 155549500 IC50 = 91.3 nM T58937 CRNC68 155549901 IC50 = 130 nM T58937 CY53JZ 155550276 IC50 = 182 nM T58937 C1L2GT 155551564 IC50 = 69.2 nM T58937 CM89BD 155555321 IC50 > 75000 nM T58937 CGF0S6 155557862 IC50 = 313 nM T58937 C17IVM 155558147 IC50 = 560 nM T58937 CP2TA6 155558730 IC50 = 47.9 nM T58937 C42VNF 155558759 IC50 = 152 nM T58937 C6VDX2 155563302 IC50 = 31.6 nM T58937 CA9P1T 155564998 IC50 > 75000 nM T58937 CIV8C4 155565435 IC50 > 75000 nM T58937 C38PJX 155566448 IC50 = 25.5 nM T58937 CB54HT 155568178 IC50 > 75000 nM T58937 D01ZHW 5283389 IC50 = 3000 nM T58937 D03TUM 16759310 IC50 = 12000 nM T58937 D07IYZ 45270374 IC50 > 10000 nM T58937 D0E1OC 16078939 IC50 = 26 nM T61622 D03SVX 5493444 IC50 = 0.4 nM T61622 D0C2EP 6324659 IC50 = 0.025 nM T61622 D0I0EG 44093 Ki = 1.7 nM T61622 D01QSG 16126898 IC50 = 1.1 nM T61622 D03XHS 12001785 IC50 = 1.4 nM T61622 D0A5SA 56591871 IC50 = 2.1 nM T61622 D0CG8S 71305058 IC50 > 200000 nM T61622 D0V3UN 64922 IC50 = 0.2 nM T61622 D00XRK 447617 IC50 > 100000 nM T61622 D04TSV 9875002 IC50 = 0.36 nM T61622 D04ZIJ 5478883 Ki = 100 nM T61622 D07PSP 5479205 Ki = 2 nM T61622 D09ELW 60594 IC50 = 0.75 nM T61622 D0J5GT 3086652 IC50 = 0.24 nM T61622 C5E9BL 3438 IC50 > 300000 nM T61622 C7A9BK 65023 IC50 > 58000 nM T61622 CDV72E 129717 IC50 = 25 nM T61622 C1EUC4 134897 IC50 = 1 nM T61622 CSO70X 147073 IC50 = 21 nM T61622 CT9HP8 157824 IC50 = 1.4 nM T61622 CFU4N8 195559 IC50 = 170 nM T61622 CFZW70 258149 IC50 > 300000 nM T61622 CEDW47 447925 IC50 = 2 nM T61622 CP7Q1V 448382 Ki = 0.7 nM T61622 C8NGY9 448772 IC50 > 500000 nM T61622 CV2P5E 454914 Ki = 1200 nM T61622 CEQ0T7 456657 IC50 = 350 nM T61622 CV58GA 460197 IC50 > 10000 nM T61622 C9QD2H 460207 IC50 > 10000 nM T61622 C19EDU 460213 IC50 > 10000 nM T61622 C0TN7S 460238 IC50 > 10000 nM T61622 CAG9E8 460240 IC50 > 10000 nM T61622 C58KVI 460241 IC50 > 10000 nM T61622 CCU6P0 460242 IC50 > 10000 nM T61622 CH7Q4G 460614 IC50 = 3400 nM T61622 C7Q0FZ 465691 IC50 = 2200 nM T61622 CKC9D6 465695 IC50 = 25 nM T61622 CIYD94 473856 IC50 = 0.52 nM T61622 CYBA13 719250 IC50 = 11000 nM T61622 CZ0U9A 837191 IC50 = 43000 nM T61622 CJI39W 3013742 IC50 = 6500 nM T61622 C50ESG 3013755 IC50 = 5200 nM T61622 CQ2P0J 3505074 IC50 = 0.7 nM T61622 CZMX32 5230731 IC50 = 1 nM T61622 CGSC72 5287532 IC50 > 50000 nM T61622 C1CZ7E 5288846 IC50 = 41 nM T61622 CO2S6C 5288847 IC50 = 56 nM T61622 C5M2JL 5327508 IC50 = 18000 nM T61622 C2ZN1E 5327509 IC50 = 600 nM T61622 CE19IN 5464201 Ki = 0.04 nM T61622 CN0VB3 6914627 IC50 = 20 nM T61622 C6JS7E 6914628 IC50 = 95 nM T61622 C80XWJ 6914629 IC50 = 90 nM T61622 CPT2S8 6914633 IC50 = 4000 nM T61622 C0MZ5V 6918046 IC50 = 2.4 nM T61622 CE4TI9 6918427 IC50 = 1.5 nM T61622 CDHA36 9802155 IC50 = 100 nM T61622 CPCF81 9806227 IC50 = 6 nM T61622 C29XJR 9809765 IC50 > 10000 nM T61622 C8KY5U 9811686 IC50 = 0.03 nM T61622 C1LZ5V 9826726 IC50 = 5.1 nM T61622 C10VHP 9826944 IC50 = 20 nM T61622 CVUF28 9833018 IC50 = 0.76 nM T61622 CZ4DQ3 9849784 IC50 = 13 nM T61622 CX0B5L 9853618 IC50 = 0.38 nM T61622 C2M5CS 9853799 IC50 = 2.4 nM T61622 C0XF3U 9871731 IC50 = 0.5 nM T61622 CRB56U 9895340 IC50 = 15 nM T61622 CZ2OT0 9896827 IC50 = 0.33 nM T61622 CC9H6V 9897236 IC50 = 4.2 nM T61622 C0Y2PH 9910816 IC50 > 100000 nM T61622 CA83IX 9916928 IC50 = 12 nM T61622 C24AWT 9917812 IC50 = 18 nM T61622 CD4BV1 9939362 IC50 = 0.067 nM T61622 C5FW7R 9939613 IC50 = 350 nM T61622 CZGY91 9961106 IC50 = 2.89 nM T61622 CW5J1V 9982638 IC50 = 1 nM T61622 C3IR4T 9985674 IC50 = 3.8 nM T61622 CS0E5K 9986272 IC50 = 1600 nM T61622 C31HKG 9986603 IC50 = 3.5 nM T61622 CLI74F 9987285 IC50 = 0.76 nM T61622 CRHX70 10006228 IC50 > 10000 nM T61622 CUJ04G 10009074 IC50 = 60.5 nM T61622 CKR2Y5 10009222 IC50 = 88 nM T61622 CG8HM9 10009841 IC50 = 14 nM T61622 CF59CE 10009918 IC50 = 3600 nM T61622 C95PVW 10010076 IC50 = 4.5 nM T61622 CHSJ03 10010399 IC50 = 14 nM T61622 CF53HQ 10010597 IC50 = 0.5 nM T61622 CLX51K 10030228 IC50 = 46 nM T61622 C3M2FR 10030516 IC50 = 17.5 nM T61622 CL79ET 10031152 IC50 = 4.2 nM T61622 CVJ8H3 10031765 IC50 = 210 nM T61622 C86JET 10032270 IC50 = 4400 nM T61622 C4XYB5 10032775 IC50 = 9.5 nM T61622 CM9CS0 10032973 IC50 = 2.6 nM T61622 CT26MZ 10033082 IC50 = 2.2 nM T61622 C48UOP 10033165 IC50 = 0.41 nM T61622 CCB2L6 10033210 IC50 = 1.1 nM T61622 C0GOV4 10046322 IC50 = 800 nM T61622 CT3N7I 10054747 IC50 = 37 nM T61622 CRYI19 10055249 IC50 = 25 nM T61622 C4NF9B 10055443 IC50 = 37 nM T61622 CY1LR3 10055510 IC50 = 69 nM T61622 CN0WO3 10055857 IC50 = 7.8 nM T61622 CIBR38 10056046 IC50 = 6.1 nM T61622 C3F9CV 10056117 IC50 = 1.3 nM T61622 CSL8G4 10056396 IC50 = 4.3 nM T61622 CPQV45 10069807 IC50 = 800 nM T61622 C9M3ZW 10070294 IC50 = 3000 nM T61622 C8BN5A 10077376 IC50 = 61 nM T61622 C8V2UW 10077648 IC50 = 22.5 nM T61622 CK1Y0M 10078377 IC50 = 34 nM T61622 C8HLY6 10078474 IC50 = 33 nM T61622 CCUX58 10078482 IC50 = 16 nM T61622 CBQ12F 10078848 IC50 = 12 nM T61622 CN32LE 10078977 IC50 = 3.8 nM T61622 C6ZS2J 10078985 IC50 = 3.1 nM T61622 C5LMR1 10078995 IC50 = 8.4 nM T61622 C36JLO 10079125 IC50 = 1.3 nM T61622 C7JXZ5 10093007 IC50 = 3000 nM T61622 C6YF4H 10099128 IC50 = 16 nM T61622 CY7P4B 10099584 IC50 > 10000 nM T61622 CG6PI7 10100513 IC50 = 66 nM T61622 CO0G6B 10100916 IC50 = 0.87 nM T61622 C18DYQ 10101068 IC50 > 1000 nM T61622 CV7SB0 10101137 IC50 = 41 nM T61622 C9WF2P 10101460 IC50 = 12 nM T61622 C65FOS 10101521 IC50 = 1.8 nM T61622 C0V7KB 10101590 IC50 = 12 nM T61622 CA2K9U 10101591 IC50 = 9.6 nM T61622 CBW6V2 10101650 IC50 = 7.9 nM T61622 CDI6R1 10101703 IC50 = 1.8 nM T61622 CI0YK5 10101718 IC50 = 3.9 nM T61622 CVX2R5 10101856 IC50 = 1.7 nM T61622 C7EAY6 10101867 IC50 = 9.2 nM T61622 COG0F3 10252386 IC50 = 130 nM T61622 C5CN2X 10254333 IC50 = 110 nM T61622 CO5EZ1 10257915 IC50 = 16 nM T61622 C3Z7GJ 10258546 IC50 = 202 nM T61622 CTSR70 10259376 IC50 = 4.3 nM T61622 C1SP5W 10326433 IC50 = 130 nM T61622 CN12SW 10326954 IC50 = 18 nM T61622 CX4R5H 10327091 IC50 = 1.1 nM T61622 CTF7L4 10327161 IC50 = 11 nM T61622 CKAL37 10327342 IC50 = 1.3 nM T61622 C9F3YP 10327393 IC50 = 9.7 nM T61622 CW0G2H 10327997 IC50 = 9.1 nM T61622 CJ9W5T 10328060 IC50 = 0.5 nM T61622 C4N8OL 10328150 IC50 = 17 nM T61622 CK5EG9 10349702 IC50 = 250 nM T61622 CUJ92M 10349779 IC50 = 39 nM T61622 CFD04C 10349956 IC50 = 1.3 nM T61622 CK39QJ 10350061 IC50 = 8.4 nM T61622 CP96LQ 10350171 IC50 = 2.4 nM T61622 CU8RI2 10350215 IC50 = 2 nM T61622 C8BFJ6 10366523 IC50 = 37 nM T61622 CQ5M4T 10370232 IC50 = 82 nM T61622 CU6O4K 10372281 IC50 = 110 nM T61622 C1EVF5 10372892 IC50 = 14 nM T61622 CB7AV4 10373009 IC50 = 40 nM T61622 C9S5AN 10373059 IC50 = 2.5 nM T61622 CBC17R 10373259 IC50 = 23 nM T61622 C2ICT0 10393697 IC50 = 2.5 nM T61622 C69KGX 10394329 IC50 = 0.16 nM T61622 CKQ25O 10394618 IC50 = 15.5 nM T61622 C0LY3Q 10394708 IC50 = 8.5 nM T61622 C1CL5Y 10394843 IC50 = 8.1 nM T61622 CZY26X 10395018 IC50 = 3 nM T61622 C8EQP4 10395167 IC50 = 4.7 nM T61622 CKON28 10395258 IC50 = 2.8 nM T61622 CALE04 10395349 IC50 = 2 nM T61622 C24LGS 10415718 IC50 = 13 nM T61622 CCM5Z3 10416850 IC50 = 5.4 nM T61622 C5V0JK 10416894 IC50 = 42 nM T61622 C03ZWQ 10416925 IC50 = 4.1 nM T61622 CC8DU9 10417164 IC50 = 1.5 nM T61622 CKDQ26 10417326 IC50 = 3.9 nM T61622 C1Y7FP 10417341 IC50 = 4 nM T61622 CCM48L 10417394 IC50 = 4.1 nM T61622 CPJ4Z1 10417593 IC50 = 11 nM T61622 CD21HS 10418066 IC50 = 11 nM T61622 CS4G3H 10436816 IC50 = 42 nM T61622 CXD53C 10439257 IC50 = 2.8 nM T61622 CP5Q4Z 10439298 IC50 = 0.36 nM T61622 CH07IE 10439438 IC50 = 0.68 nM T61622 CY53UB 10439575 IC50 = 17 nM T61622 CDL80M 10439577 IC50 = 0.6 nM T61622 CRBT74 10439647 IC50 = 5 nM T61622 C5MV2B 10439855 IC50 = 2.6 nM T61622 CLV15O 10440018 IC50 = 33 nM T61622 C8HZB4 10440125 IC50 = 6 nM T61622 CVZ56U 10440267 IC50 = 3.3 nM T61622 C6JB5T 10458380 IC50 = 120 nM T61622 CE8GQ3 10461191 IC50 = 94 nM T61622 CP3GK9 10461457 IC50 = 11 nM T61622 CT2XM5 10461538 IC50 = 18.5 nM T61622 C0OH5D 10461649 IC50 = 25 nM T61622 CH1PX0 10461792 IC50 = 93 nM T61622 C9HQ3X 10462138 IC50 = 9.4 nM T61622 CWY05N 10462142 IC50 = 0.48 nM T61622 C9J0YI 10462166 IC50 = 33 nM T61622 CW8JQ3 10462664 IC50 = 1.6 nM T61622 CEKA23 10462689 IC50 = 0.2 nM T61622 CO0YM8 10462909 IC50 = 6.3 nM T61622 C70BDS 10463080 IC50 = 21 nM T61622 C3G9ZI 10475887 IC50 = 300 nM T61622 CD1O4Z 10483146 IC50 = 12 nM T61622 CK2T0P 10483414 IC50 = 13 nM T61622 CF0J4D 10484665 IC50 = 3.9 nM T61622 CXNS04 10484822 IC50 = 0.72 nM T61622 CK9F8X 10484900 IC50 = 0.16 nM T61622 CUBX08 10484999 IC50 = 0.8 nM T61622 C0JKB4 10485007 IC50 = 12 nM T61622 C4Y8BX 10485092 IC50 = 8.4 nM T61622 CC1X4N 10485248 IC50 = 13 nM T61622 C6YQG3 10485297 IC50 = 9.4 nM T61622 CG9R2A 10485490 IC50 = 3.3 nM T61622 C9XHP2 10485494 IC50 = 4.3 nM T61622 C76WLB 10485512 IC50 = 230 nM T61622 C2L8HV 10531945 IC50 = 16 nM T61622 CKP6D0 10556249 IC50 = 41000 nM T61622 CX3QN9 10627507 IC50 = 27000 nM T61622 CO87HB 10627883 IC50 = 8.5 nM T61622 CL0G3V 10699067 IC50 = 400 nM T61622 CC81FU 10699555 IC50 = 41 nM T61622 CYE97S 10746764 IC50 = 220 nM T61622 CY62GO 10770128 IC50 = 5200 nM T61622 CIG63W 10770392 IC50 = 31 nM T61622 C89LKM 10770530 IC50 = 38 nM T61622 CGWZ23 10794358 IC50 = 29 nM T61622 CYBH12 11123690 IC50 = 220 nM T61622 C27OAY 11204336 IC50 = 7 nM T61622 CMR0S9 11214666 IC50 = 54 nM T61622 CR9I4L 11227351 IC50 = 0.42 nM T61622 CEW9L6 11228293 Ki > 20000 nM T61622 CF9X3W 11273357 IC50 = 120 nM T61622 C9W2NY 11274374 Ki > 4000 nM T61622 C4E9PK 11280673 IC50 = 27000 nM T61622 C5I9RP 11289532 IC50 = 30000 nM T61622 C19BEF 11330998 IC50 = 0.29 nM T61622 C2LFN6 11342476 IC50 > 50000 nM T61622 CR0TE8 11342515 IC50 > 50000 nM T61622 C76RIA 11365730 IC50 = 800 nM T61622 C6H1UP 11375292 IC50 = 12 nM T61622 C5QL8O 11376341 IC50 > 50000 nM T61622 CDF21W 11387864 IC50 = 3.2 nM T61622 CU9OR7 11388049 IC50 = 9 nM T61622 CHX8E5 11410816 IC50 > 10000 nM T61622 CIPA26 11410903 IC50 > 50000 nM T61622 CH4PV3 11420856 IC50 = 61 nM T61622 C84MEW 11421906 IC50 > 50000 nM T61622 C1V7WT 11422288 IC50 = 0.18 nM T61622 C3E1DQ 11445043 IC50 = 4000 nM T61622 CS05AN 11456311 IC50 = 17 nM T61622 C95NIM 11504581 IC50 = 141 nM T61622 CG9R2S 11505504 IC50 = 23 nM T61622 CDB52K 11516368 IC50 = 18000 nM T61622 C3P6ZU 11516577 IC50 = 93400 nM T61622 CYIV63 11517020 IC50 = 57600 nM T61622 CW68BJ 11518143 IC50 = 170 nM T61622 C18CGE 11518439 IC50 = 770 nM T61622 CPK79W 11532880 IC50 = 20800 nM T61622 CS8NW6 11578126 IC50 = 0.2 nM T61622 C3LW2D 11632240 IC50 = 7600 nM T61622 CEM04T 11641967 IC50 = 0.47 nM T61622 C14JYI 11668187 IC50 = 42300 nM T61622 CPU08S 11671739 IC50 = 0.16 nM T61622 CW1BU5 11705154 IC50 = 2700 nM T61622 CGE50S 11757267 Ki = 73600 nM T61622 C93VXK 11758460 IC50 = 11 nM T61622 CJE61H 11765063 IC50 = 85 nM T61622 CHC20N 11765175 IC50 = 53 nM T61622 C6K7ZT 11765209 IC50 = 1.6 nM T61622 CQ9B3X 11765277 IC50 = 46 nM T61622 C0D3MN 11765479 IC50 = 8.5 nM T61622 CW2D4B 11765498 IC50 = 6.8 nM T61622 C0FP7L 11765780 IC50 = 1.5 nM T61622 CPQ2Z1 11765860 IC50 = 5.9 nM T61622 CW4RP0 11840980 IC50 = 23 nM T61622 CHD3B0 11949623 IC50 = 90 nM T61622 CPT14W 11962165 IC50 = 364 nM T61622 CLP92O 11963435 IC50 = 3 nM T61622 C8NY4Q 11963439 IC50 = 4000 nM T61622 CQL8U4 11963547 IC50 = 27 nM T61622 CGN27B 11963989 IC50 = 3.6 nM T61622 C4C2RS 11993712 IC50 = 1200 nM T61622 C2JP6D 12001701 IC50 = 0.31 nM T61622 CV1IS7 12001783 IC50 = 0.33 nM T61622 C2HV4P 12001784 IC50 = 0.18 nM T61622 C2QAW5 12001786 IC50 = 0.28 nM T61622 CQKJ25 12001869 IC50 = 0.27 nM T61622 CF0C8W 12001871 IC50 = 4.1 nM T61622 CHE5V2 12001872 IC50 = 3.9 nM T61622 C2F1JZ 12001873 IC50 = 1.39 nM T61622 CK7CQ0 12001952 IC50 = 0.41 nM T61622 CM68CQ 12001953 IC50 = 0.4 nM T61622 C17AVT 12001954 IC50 = 0.18 nM T61622 CS5BA8 12001955 IC50 = 0.15 nM T61622 CL6OY0 12001956 IC50 = 2.17 nM T61622 CP10LA 12002034 IC50 = 0.31 nM T61622 CC7BS3 12002035 IC50 = 0.56 nM T61622 CG4MW9 13105154 Ki = 1.2 nM T61622 CM2SE4 13334744 Ki = 500000 nM T61622 CX1H4I 13384509 IC50 = 3467.37 nM T61622 C2L8HS 13384512 IC50 = 1000 nM T61622 C87OJL 13384515 IC50 = 76 nM T61622 CWQ65F 13384518 IC50 = 151.36 nM T61622 C9MOQ8 13384519 IC50 > 100000 nM T61622 C3UV1C 13384520 IC50 > 100000 nM T61622 C52BGR 13384530 IC50 = 140 nM T61622 CZK2M8 13384541 IC50 = 300 nM T61622 C8EY5X 13384551 IC50 = 10000 nM T61622 C3G4AI 13384553 IC50 = 110 nM T61622 CBN1H5 13385305 IC50 = 140 nM T61622 C3QS2P 13385307 IC50 = 63 nM T61622 C5T7WM 13385517 IC50 = 5.7 nM T61622 CY71GE 13385537 Ki = 0.064 nM T61622 C6L0JM 13420901 IC50 = 80 nM T61622 CGS1B8 13420917 IC50 = 1500 nM T61622 C5W8PN 13420933 IC50 = 6400 nM T61622 C94AZE 13420949 IC50 = 16000 nM T61622 CT8D3A 13605353 IC50 = 28 nM T61622 C58IRJ 13752786 IC50 = 316.23 nM T61622 C1XAF6 13851544 IC50 = 0.5 nM T61622 CTIO41 13852880 IC50 = 45 nM T61622 C7HW1F 13876183 IC50 = 120.23 nM T61622 C4XJL9 13877753 IC50 = 10 nM T61622 CK3H0B 13877755 IC50 = 10 nM T61622 C4W9HE 13877757 IC50 = 50 nM T61622 CA84WS 13877759 IC50 = 150 nM T61622 CN75ZC 13877761 IC50 = 50 nM T61622 CYEW26 13877763 IC50 = 400 nM T61622 CL9J2N 13877765 IC50 = 25 nM T61622 CSB87X 13877767 IC50 = 200 nM T61622 CE4V7Y 13877770 IC50 = 400 nM T61622 CBJ1D8 13877773 IC50 = 1.5 nM T61622 CXG82M 13877776 IC50 = 2 nM T61622 C67VDF 13877779 IC50 = 5 nM T61622 CS48WF 13877788 IC50 = 3 nM T61622 C1O6BV 13877790 IC50 = 4 nM T61622 C2XB6M 13877792 IC50 = 2000 nM T61622 CNE1J3 13877796 IC50 = 4 nM T61622 C07JKH 13877798 IC50 = 5 nM T61622 CP93KR 13877801 IC50 = 10 nM T61622 C1R8ZJ 13877805 IC50 = 8.5 nM T61622 C98NXF 13877810 IC50 = 2 nM T61622 CB56QG 13877812 IC50 = 25 nM T61622 CL3DV4 13877814 IC50 = 40 nM T61622 CWV29D 13877841 IC50 = 5.5 nM T61622 C3W0DT 13877842 IC50 = 50 nM T61622 CWF8Y6 13877844 IC50 = 20 nM T61622 CN7I6H 13877845 IC50 = 1 nM T61622 C9QW2E 13877847 IC50 = 30 nM T61622 CMJ7W0 13877849 IC50 = 20 nM T61622 C7HBD1 13877850 IC50 = 0.8 nM T61622 CF53VP 13877852 IC50 = 35 nM T61622 CFUS31 13877853 IC50 = 15 nM T61622 C4BA9O 13884399 IC50 = 2600 nM T61622 C7TL1W 13891064 IC50 = 2400 nM T61622 CF2WL1 13891066 IC50 = 3800 nM T61622 CS58ZN 13891087 IC50 = 5500 nM T61622 CH0RM3 13891089 IC50 = 4200 nM T61622 C5LAD6 13891091 IC50 = 4100 nM T61622 C0Q7AE 13891093 IC50 = 4800 nM T61622 C8ATQ0 13891095 IC50 = 5200 nM T61622 C90SXY 13891097 IC50 = 2400 nM T61622 CQ8E4J 13891099 IC50 = 1800 nM T61622 C0MB1C 13891101 IC50 = 3200 nM T61622 CWGF24 13891103 IC50 = 1600 nM T61622 C61ERQ 13891128 IC50 = 7.6 nM T61622 C18SHD 13891130 IC50 = 7.6 nM T61622 CRQX06 13891132 IC50 = 9.1 nM T61622 CG51HL 13891136 IC50 = 6 nM T61622 C2R6FE 13891138 IC50 = 23 nM T61622 C7SFT5 13891140 IC50 = 76 nM T61622 C2Q8OF 13891142 IC50 = 140 nM T61622 C1G5QT 13891144 IC50 = 14 nM T61622 C7P5VT 13891146 IC50 = 340 nM T61622 C6ONC9 13892812 IC50 = 15 nM T61622 CPME08 13892814 IC50 = 4 nM T61622 C1Z2WT 13892816 IC50 = 6.5 nM T61622 CC02OQ 13892818 IC50 = 4 nM T61622 CPY5V1 13892820 IC50 = 10 nM T61622 CL7F6V 13892823 IC50 = 2.5 nM T61622 C1EVA5 13892826 IC50 = 2 nM T61622 C7U4VQ 13892829 IC50 = 40 nM T61622 CXZD08 13892831 IC50 = 9 nM T61622 CPNX91 13892833 IC50 = 70 nM T61622 C3DVZ7 13892842 IC50 = 4 nM T61622 CGV3S1 13892844 IC50 = 30 nM T61622 C4OTI6 13892848 IC50 = 40 nM T61622 CH6BL0 13892851 IC50 = 20 nM T61622 CH74DM 13892859 IC50 = 60 nM T61622 CR5YP6 13892870 IC50 = 100 nM T61622 CZM1P4 13892874 IC50 = 300 nM T61622 CMD3I2 13892876 IC50 = 75 nM T61622 CFH9I0 13892886 IC50 = 3 nM T61622 CPE37U 13892914 IC50 = 3 nM T61622 CSUH30 13892915 IC50 = 3.5 nM T61622 CYX98H 13892917 IC50 = 5 nM T61622 CPVA72 13893166 IC50 = 81 nM T61622 C5UYG4 13893168 IC50 = 520 nM T61622 CSM46O 13893200 IC50 = 700 nM T61622 CF9UM7 13893236 IC50 = 1500 nM T61622 C6NK2L 13893238 IC50 = 2000 nM T61622 C10WJF 13893290 Ki = 120 nM T61622 C6H9VT 13893292 Ki = 7 nM T61622 C8GTW0 13893294 Ki = 12000 nM T61622 C2JBM6 13893303 Ki = 16000 nM T61622 CVA0E1 13893305 Ki = 1200 nM T61622 CE74TY 13913914 IC50 = 11 nM T61622 CPT61D 13913919 IC50 = 130 nM T61622 CK2U9Z 13913924 IC50 = 24 nM T61622 C27KVE 13913931 IC50 = 25 nM T61622 CLY0G9 13913938 IC50 = 66 nM T61622 C3VPN5 13996493 IC50 = 1.7 nM T61622 CVS52D 14014862 IC50 = 1500 nM T61622 C36LGM 14014863 IC50 = 2300 nM T61622 C65ZLD 14014864 IC50 = 2100 nM T61622 CJY0L3 14104733 IC50 = 4000 nM T61622 CNF53G 14104735 IC50 = 250 nM T61622 C6EP4Y 14212866 Ki = 1 nM T61622 CGT04D 14212875 IC50 = 4000 nM T61622 C0IA5P 14212882 IC50 = 4000 nM T61622 CEL8C5 14212884 IC50 = 350 nM T61622 CHF0V5 14212887 IC50 = 200 nM T61622 C93LGV 14212890 IC50 = 10 nM T61622 CCH9A1 14212893 IC50 = 11 nM T61622 CB2CJ1 14212896 IC50 = 1.5 nM T61622 CKU7T2 14212900 IC50 = 70 nM T61622 C29VYB 14212902 IC50 = 95 nM T61622 CDKL37 14212904 IC50 = 0.6 nM T61622 C1WYB0 14212906 IC50 = 0.3 nM T61622 CZ3FP0 14212909 IC50 = 2 nM T61622 C8MD5L 14212911 IC50 = 5 nM T61622 CW8S9Z 14212913 IC50 = 1.5 nM T61622 CYFP27 14212917 IC50 = 0.5 nM T61622 C8LP3G 14212923 IC50 = 1 nM T61622 C12TLP 14212927 IC50 = 1.5 nM T61622 CQZ50T 14212929 IC50 = 1 nM T61622 CM4W5V 14212932 IC50 = 200 nM T61622 C4B7KN 14212937 IC50 = 1 nM T61622 CFA34W 14212939 IC50 = 1 nM T61622 C48TGH 14212941 IC50 = 2 nM T61622 CK3I2C 14212944 IC50 = 0.75 nM T61622 CC74MQ 14212950 IC50 = 0.7 nM T61622 C3V8DH 14212952 IC50 = 0.25 nM T61622 C9AN3J 14212954 IC50 = 0.2 nM T61622 CI7YM2 14212956 IC50 = 1.5 nM T61622 C0WFN2 14212958 IC50 = 1 nM T61622 CCR81U 14212962 IC50 = 2.4 nM T61622 C6YN4R 14212965 IC50 = 50 nM T61622 C69KMP 14212967 IC50 = 2 nM T61622 CTE56K 14212970 IC50 = 0.6 nM T61622 C7EV8X 14212972 IC50 = 1.5 nM T61622 CI3BF0 14212975 IC50 = 4 nM T61622 C1P7WM 14212977 IC50 = 0.5 nM T61622 CYC74N 14212980 IC50 = 1.1 nM T61622 CVR6C8 14212983 IC50 = 10 nM T61622 C74VQT 14213025 IC50 = 0.5 nM T61622 CWD7H8 14213027 IC50 = 0.42 nM T61622 CUT9D4 14213029 IC50 = 0.65 nM T61622 CQ96PH 14213031 IC50 = 0.55 nM T61622 C1V5AG 14213033 IC50 = 0.35 nM T61622 CV9NQ4 14213034 IC50 = 14 nM T61622 C4GQX5 14213036 IC50 = 2 nM T61622 CM0J9E 14213038 IC50 = 0.76 nM T61622 C9OEX3 14213040 IC50 = 0.82 nM T61622 CMYX89 14213042 IC50 = 2.1 nM T61622 C9M1GH 14213044 IC50 = 1.6 nM T61622 CG9X0Y 14213051 IC50 = 2.6 nM T61622 C61LCY 14213054 IC50 = 0.94 nM T61622 CL1XV9 14301580 IC50 = 2.1 nM T61622 C3JWD2 14301583 IC50 = 6.3 nM T61622 C93EGF 14301584 IC50 = 5.5 nM T61622 C43ZOE 14301589 IC50 = 4.2 nM T61622 CZJ1T5 14478735 IC50 = 0.4 nM T61622 CHY31B 14590920 IC50 = 0.29 nM T61622 CU4Z8A 14654517 IC50 = 4.7 nM T61622 C0JQ3A 14654520 IC50 = 8.8 nM T61622 C08BSE 14654523 IC50 = 2.8 nM T61622 C0HK9Q 14654526 IC50 = 9.2 nM T61622 C31PFQ 14654529 IC50 = 0.84 nM T61622 CZT2W7 14654532 IC50 = 1 nM T61622 C81ODH 14654535 IC50 = 1.3 nM T61622 CWV0H1 14654538 IC50 = 0.7 nM T61622 C82JEL 14654541 IC50 = 21 nM T61622 CQOG71 14654544 IC50 = 26 nM T61622 C4OM8X 14654547 IC50 = 3.1 nM T61622 CP0W3J 14654550 IC50 = 11 nM T61622 C1PUV7 14654553 IC50 = 1.4 nM T61622 C5J6OR 14654556 IC50 = 0.71 nM T61622 CQ84AW 14654559 IC50 = 0.32 nM T61622 C9T5JC 14654562 IC50 = 0.89 nM T61622 C1ALY0 14654567 IC50 = 8 nM T61622 C8ULZ1 14696176 IC50 = 32 nM T61622 CCYQ36 14696179 IC50 = 448 nM T61622 C9TVY8 14731929 IC50 = 10 nM T61622 CC9K0V 14771989 IC50 = 0.85 nM T61622 C14TXU 14775317 IC50 = 1100 nM T61622 CD81UJ 14775318 IC50 > 100000 nM T61622 CNI4Z8 14787980 IC50 = 30 nM T61622 C5NC0Z 14787982 IC50 = 2.7 nM T61622 CN8OL5 14787985 IC50 = 0.2 nM T61622 CN8IL9 14787990 IC50 = 0.3 nM T61622 C80YWK 14787993 IC50 = 78 nM T61622 C0LT8Z 14787995 IC50 = 0.4 nM T61622 C29JDS 14787997 IC50 = 0.6 nM T61622 C58KHQ 14787999 IC50 = 0.6 nM T61622 CMYQ89 14788001 IC50 = 0.3 nM T61622 C20TVK 14788003 IC50 = 41 nM T61622 CN58IE 14788005 IC50 = 212 nM T61622 CGR4W7 14788007 IC50 = 64 nM T61622 CK34RF 14803030 IC50 = 0.33 nM T61622 CI8MO5 14803040 IC50 = 1.6 nM T61622 CY84WR 14803056 IC50 = 0.29 nM T61622 CIA54G 14803060 IC50 = 0.43 nM T61622 C5RH4S 14803068 IC50 = 0.29 nM T61622 CSQD49 14803074 IC50 = 0.32 nM T61622 C73NXE 14850260 IC50 = 100 nM T61622 CWYK87 14861426 IC50 = 23 nM T61622 C17NYD 14861476 IC50 = 10000 nM T61622 C01KUS 14861671 IC50 = 130 nM T61622 C4GS1X 14861674 IC50 = 4 nM T61622 C3N0GZ 14861675 IC50 = 0.79 nM T61622 CUB43M 14861679 IC50 = 0.28 nM T61622 CIDF93 14861680 IC50 = 0.28 nM T61622 CE29TK 14887165 IC50 = 5.5 nM T61622 CJO10Z 14887166 IC50 > 20000 nM T61622 C02NGW 14887167 IC50 = 280 nM T61622 CJ8R0O 14887174 IC50 = 8 nM T61622 CHIC86 14887175 IC50 = 2.5 nM T61622 C56EWA 14887177 IC50 = 4400 nM T61622 C2LRD8 14887179 IC50 = 40 nM T61622 CT4V6C 14887181 IC50 = 1.3 nM T61622 C4UA0C 14887183 IC50 = 1.9 nM T61622 C6JF8N 14887185 IC50 = 10 nM T61622 CH0VA6 14887187 IC50 = 24 nM T61622 CZ17YD 14887189 IC50 = 275 nM T61622 C5N4PO 14887191 IC50 = 8.5 nM T61622 C26HVF 14887192 IC50 = 3.3 nM T61622 CAKS64 14887194 IC50 = 14 nM T61622 C5LC4F 14887196 IC50 = 155 nM T61622 CGRF98 14887198 IC50 = 7.7 nM T61622 CLQA57 14887200 IC50 = 14 nM T61622 C4LK1Q 14990021 IC50 = 2.7 nM T61622 C8KU7J 14990024 IC50 = 3.61 nM T61622 C6W1JK 14990027 IC50 = 0.59 nM T61622 C7WYD5 14990028 IC50 = 0.5 nM T61622 C84EIU 14990029 IC50 = 0.54 nM T61622 CE2W9P 14990030 IC50 = 0.2 nM T61622 CO21PC 14991474 IC50 = 2.2 nM T61622 CD59EM 14991475 IC50 = 110 nM T61622 CRHY93 14991481 IC50 = 4.7 nM T61622 CZC10K 14991482 IC50 = 6 nM T61622 CZ07LT 14991483 IC50 = 2.7 nM T61622 C9O8WX 14991484 IC50 = 1.7 nM T61622 CCJ1D3 14991485 IC50 = 11 nM T61622 C6NYH1 14991486 IC50 = 12 nM T61622 CE8S4T 14991487 IC50 = 28 nM T61622 C1AFN8 14991488 IC50 = 2.8 nM T61622 C2VXN4 14991489 IC50 = 1.3 nM T61622 CQ2M8H 14991490 IC50 = 28 nM T61622 CA9O0P 14991491 IC50 = 67 nM T61622 C53SJC 14991492 IC50 = 3.2 nM T61622 CYB5F1 14991493 IC50 = 2.4 nM T61622 C8U7EM 14991494 IC50 = 1.5 nM T61622 C5VFB0 14991495 IC50 = 5 nM T61622 C7YWI6 14991496 IC50 = 2.7 nM T61622 C4T9ZI 14991497 IC50 = 2.5 nM T61622 CRS6M0 14991498 IC50 = 1.4 nM T61622 C1TW8N 14991499 IC50 = 2.4 nM T61622 CM9W8L 14991500 IC50 = 0.9 nM T61622 CS3B7J 14991501 IC50 = 1.5 nM T61622 CGP3D5 14991502 IC50 = 1.8 nM T61622 C5Z1DK 14991512 IC50 = 2.9 nM T61622 C5C7SL 14991513 IC50 = 290 nM T61622 C7V5TK 14991514 IC50 = 2.5 nM T61622 C1HFQ7 14991515 IC50 = 57 nM T61622 C1JOU3 14991516 IC50 = 17 nM T61622 CTP18H 14991517 IC50 = 1 nM T61622 C7AQE6 14991518 IC50 = 1.3 nM T61622 C3CV8Z 14991520 IC50 = 0.9 nM T61622 COA8R4 14991521 IC50 = 2.1 nM T61622 CLZY32 14991525 IC50 = 61 nM T61622 C1ZA3W 15016694 IC50 = 20 nM T61622 CFQ2W6 15018067 IC50 = 0.9 nM T61622 CE12CX 15018069 IC50 = 0.7 nM T61622 C5N2GB 15021438 IC50 = 8.9 nM T61622 C2ARE4 15021442 IC50 = 16 nM T61622 CVU17T 15109734 IC50 = 70 nM T61622 CA01IK 15109735 IC50 = 240 nM T61622 C9O2FB 15109747 IC50 = 0.53 nM T61622 CMYL49 15109749 IC50 = 8.5 nM T61622 C32JEK 15109751 IC50 = 5.4 nM T61622 C6O2NJ 15109752 IC50 = 4.1 nM T61622 CK32FJ 15109753 IC50 = 5.1 nM T61622 C2EY5K 15109754 IC50 = 5.4 nM T61622 C1FS8W 15109755 IC50 = 19.5 nM T61622 C8J3MU 15109759 IC50 = 8 nM T61622 CP02TJ 15109762 IC50 = 0.28 nM T61622 CHC89K 15109764 IC50 = 0.41 nM T61622 C8NE3W 15109767 IC50 = 0.58 nM T61622 CI41XT 15126555 IC50 = 0.8 nM T61622 CBTS23 15126556 IC50 = 0.4 nM T61622 C48BLM 15126557 IC50 = 0.23 nM T61622 CO17XG 15126560 IC50 = 0.36 nM T61622 C6K2ST 15126561 IC50 = 0.31 nM T61622 CK41QJ 15126568 IC50 = 0.35 nM T61622 CJE92F 15126569 IC50 = 0.25 nM T61622 CW8N4M 15126570 IC50 = 1.17 nM T61622 C72QTB 15126573 IC50 = 0.3 nM T61622 CJQ0O6 15126581 IC50 = 2.46 nM T61622 C8SF1J 15126582 IC50 = 0.35 nM T61622 C1SKE6 15126583 IC50 = 0.1 nM T61622 CH1CD3 15126584 IC50 = 0.92 nM T61622 C2TZV3 15126585 IC50 = 3.55 nM T61622 C1KGM8 15126586 IC50 = 0.23 nM T61622 CCR5U3 15172668 IC50 = 198 nM T61622 CU32YJ 15172669 IC50 = 240 nM T61622 CY46CT 15172670 IC50 = 3310 nM T61622 CEA4G3 15172671 IC50 = 124 nM T61622 C7Y0XF 15172672 IC50 = 708 nM T61622 CC45LR 15172673 IC50 = 81 nM T61622 C12TXC 15172674 IC50 = 39 nM T61622 CAQ41C 15172675 IC50 = 392 nM T61622 CV0E8S 15172676 IC50 = 206 nM T61622 C30HGJ 15172677 IC50 = 41 nM T61622 CMF68H 15172678 IC50 = 33 nM T61622 CAU5Z7 15172679 IC50 = 31 nM T61622 CREZ71 15172680 IC50 = 145 nM T61622 CO6EQ8 15172681 IC50 = 39 nM T61622 CL8E1W 15172682 IC50 = 207 nM T61622 C2TG9K 15172683 IC50 = 678 nM T61622 CP70YC 15172685 IC50 = 396 nM T61622 C87HRQ 15172686 IC50 = 1290 nM T61622 C8TQ3A 15172687 IC50 = 314 nM T61622 C9PS0O 15172688 IC50 = 359 nM T61622 CZ5GQ2 15172689 IC50 = 37 nM T61622 CL6V1K 15172736 IC50 = 130 nM T61622 CTO83Y 15172737 IC50 = 1000 nM T61622 C2QVT7 15172738 IC50 = 2700 nM T61622 CG8UI1 15172739 IC50 = 340 nM T61622 CZE60A 15172740 IC50 = 85 nM T61622 CG3B2V 15172741 IC50 = 1000 nM T61622 C21DNP 15172742 IC50 = 750 nM T61622 CAK20N 15172783 IC50 = 1 nM T61622 C4VQD7 15172788 IC50 = 1.2 nM T61622 C28REY 15172790 IC50 = 1.1 nM T61622 CC18XP 15172791 IC50 = 160 nM T61622 CXM0D5 15172792 IC50 = 290 nM T61622 CLF92V 15172793 IC50 = 130 nM T61622 CCJ68U 15172794 IC50 = 130 nM T61622 CWL0X6 15172795 IC50 = 770 nM T61622 C5MN6D 15172796 IC50 = 780 nM T61622 CAV6G9 15172797 IC50 = 4300 nM T61622 C73BRG 15172798 IC50 = 15 nM T61622 CM4J2Q 15172799 IC50 = 130 nM T61622 CA1N0K 15172800 IC50 > 1000 nM T61622 CU5SB4 15172801 IC50 = 5.5 nM T61622 CQP2U4 15172802 IC50 = 12 nM T61622 CNAG29 15172803 IC50 = 25 nM T61622 CC3I6T 15172804 IC50 = 24 nM T61622 C29LSX 15172805 IC50 = 44 nM T61622 CQTB18 15172806 IC50 = 18 nM T61622 C62OWJ 15172807 IC50 = 1.3 nM T61622 C8LUK7 15172808 IC50 = 31 nM T61622 CAO9S2 15172809 IC50 = 1100 nM T61622 CVD4N6 15172810 IC50 = 1.8 nM T61622 C95PHD 15172811 IC50 = 160 nM T61622 CPL64V 15177204 IC50 = 615 nM T61622 CK5HS1 15235163 IC50 = 1.3 nM T61622 C3ANU9 15601552 IC50 = 20000 nM T61622 CD72VG 15601554 IC50 = 450 nM T61622 C7J4BI 15601556 IC50 = 1000 nM T61622 CA84JD 15601558 IC50 = 55000 nM T61622 CTHX04 15601578 IC50 = 1500 nM T61622 C38GTX 15601586 IC50 = 170 nM T61622 C4XVE3 15601588 IC50 = 150 nM T61622 CR8O9D 15601590 IC50 = 1500 nM T61622 C86SRO 15601596 IC50 = 19 nM T61622 CU07EY 15615049 IC50 = 52 nM T61622 CM9CY0 15615051 IC50 = 28 nM T61622 CEJ4D0 15630819 IC50 = 500 nM T61622 CO40WP 15630829 IC50 = 5 nM T61622 CY98MB 15648564 IC50 = 40000 nM T61622 C7GU6X 15648565 IC50 > 1000 nM T61622 C25TVR 15659150 IC50 = 26 nM T61622 CNU67M 15659151 IC50 = 95 nM T61622 CI7PJ2 15659153 IC50 > 1000 nM T61622 CTH81G 15659154 IC50 = 210 nM T61622 CO7M1R 15659155 IC50 = 180 nM T61622 CKWQ36 15659156 IC50 = 633 nM T61622 C7FH1I 15659157 IC50 = 95 nM T61622 C8M1HL 15659158 IC50 > 1000 nM T61622 CP0H4W 15659159 IC50 = 656 nM T61622 CR5S2I 15659160 IC50 = 1000 nM T61622 CKFV51 15659161 IC50 = 500 nM T61622 CWG5J0 15659162 IC50 = 74 nM T61622 CSU4K5 15659163 IC50 = 310 nM T61622 CO6ZN8 15659164 IC50 = 936 nM T61622 C0SFK1 15659165 IC50 = 516 nM T61622 C5ZT0J 15659167 IC50 = 0.25 nM T61622 CQO94A 15659169 IC50 = 0.1 nM T61622 C70UKX 15659170 IC50 = 0.21 nM T61622 CEQ1C8 15659172 IC50 = 0.22 nM T61622 CWQ0N7 15659173 IC50 = 0.52 nM T61622 CSAZ54 15659174 IC50 = 0.18 nM T61622 CPSQ76 15659176 IC50 = 0.17 nM T61622 C0OTP4 15659178 IC50 = 13 nM T61622 CD61SU 15659179 IC50 = 0.23 nM T61622 C61BDQ 15659181 IC50 = 1.4 nM T61622 C74KRL 15659182 IC50 = 35 nM T61622 CW3PZ6 15659183 IC50 = 5.3 nM T61622 CA1PD5 15659185 IC50 = 0.44 nM T61622 CP30KG 15659186 IC50 = 1.5 nM T61622 CIB4C3 15659188 IC50 = 2.1 nM T61622 CN72WE 15673234 IC50 = 904 nM T61622 CX18HV 15673236 IC50 = 58 nM T61622 CI0RN8 15673248 IC50 = 288 nM T61622 C2M4OL 15673249 IC50 = 305 nM T61622 C8NVS3 15673251 IC50 = 92 nM T61622 C5ER7D 15673252 IC50 = 161 nM T61622 C2K7SP 15673253 IC50 = 29 nM T61622 CRS03P 15673260 IC50 = 40 nM T61622 C03GLK 15673261 IC50 = 29 nM T61622 CS3TW2 15673262 IC50 = 19 nM T61622 C6ZOT5 15673263 IC50 = 9.4 nM T61622 C06NIQ 15673264 IC50 = 20 nM T61622 CYZ14J 15673265 IC50 = 34 nM T61622 C1JET7 15673267 IC50 = 88 nM T61622 C7ED4P 15673269 IC50 = 77 nM T61622 CFC02Z 15689668 IC50 = 610 nM T61622 CQB7H4 15689669 IC50 = 9200 nM T61622 CGT5F3 15689670 IC50 = 590 nM T61622 CI60CU 15689671 IC50 = 14000 nM T61622 CEU8H2 15689672 IC50 > 20000 nM T61622 CTY6N4 15689673 IC50 = 650 nM T61622 CHMN49 15689674 IC50 > 20000 nM T61622 CB9C2P 15689675 IC50 = 56 nM T61622 C87TQR 15714045 IC50 = 0.37 nM T61622 CJ6SC9 15714072 IC50 = 0.13 nM T61622 CR70TK 15714121 IC50 = 1.3 nM T61622 CY6W5Q 15725560 IC50 = 134 nM T61622 CJU46K 15725561 IC50 = 5910 nM T61622 CBQE92 15725562 IC50 = 21 nM T61622 C9DJL5 15725567 IC50 > 20000 nM T61622 CV5P4G 15725568 IC50 = 2040 nM T61622 CSLQ07 15725569 IC50 = 1730 nM T61622 C6FBA4 15755386 IC50 = 16 nM T61622 CA7E4W 15755387 IC50 = 10 nM T61622 CJU13X 15755388 IC50 = 92 nM T61622 C4Q0CI 15755390 IC50 = 19 nM T61622 C2JI4D 15755391 IC50 = 2.1 nM T61622 CT0LM5 15755392 IC50 = 33 nM T61622 C57OAI 15755394 IC50 = 200 nM T61622 CRI98Z 15755395 IC50 = 0.7 nM T61622 CRK61C 15755396 IC50 = 120 nM T61622 CEWP83 15755398 IC50 = 120 nM T61622 C3V1HE 15755399 IC50 = 25 nM T61622 CXN3K0 15755400 IC50 = 27 nM T61622 CV14TN 15755402 IC50 = 0.47 nM T61622 CR3V6J 15755403 IC50 = 150 nM T61622 CPBY63 15924453 IC50 = 0.65 nM T61622 CW7DP0 15924500 IC50 = 4.5 nM T61622 C1Y7ER 15981115 IC50 = 0.4 nM T61622 CMD07X 15981118 IC50 = 1.9 nM T61622 CW3UJ1 15981153 IC50 = 260 nM T61622 C0D2SA 15981185 IC50 = 210 nM T61622 C8G4RJ 15981186 IC50 = 0.79 nM T61622 CIC7E3 16036820 IC50 = 7.762 nM T61622 CMZU26 16043268 IC50 = 7 nM T61622 C0QAD8 16050550 IC50 = 53300 nM T61622 CPZY01 16066132 IC50 = 10.23 nM T61622 CIV72W 16086657 IC50 = 36 nM T61622 C2HMT5 16113206 IC50 = 6900 nM T61622 CX39UL 16113753 IC50 = 44000 nM T61622 CL38QC 16220179 IC50 = 15 nM T61622 C4Q2WZ 16717887 IC50 = 0.48 nM T61622 CYQ34L 16717890 IC50 = 6.2 nM T61622 COIQ32 16717938 IC50 = 0.61 nM T61622 C3B8DO 16717939 IC50 = 0.52 nM T61622 C2VIO1 16717995 IC50 = 1.8 nM T61622 CI7Z6F 16741239 IC50 = 2700 nM T61622 C2V1ET 18654288 IC50 = 34 nM T61622 C5HFI2 19039521 IC50 = 0.9 nM T61622 CTA18D 21968125 IC50 = 0.5 nM T61622 C35RJC 22126742 IC50 = 50000 nM T61622 CZ93IM 22874640 IC50 = 8 nM T61622 C61LKZ 23277665 IC50 = 0.4 nM T61622 CQSB59 23586140 IC50 = 37 nM T61622 CJG25Z 23624691 IC50 = 92 nM T61622 C81OBN 23624692 IC50 = 50 nM T61622 C2D8YL 23624857 IC50 = 0.6 nM T61622 C95PVE 23624858 IC50 = 3 nM T61622 C7VI9O 23624859 IC50 = 2 nM T61622 CA1O3T 23624860 IC50 = 4 nM T61622 CGTU49 23624861 IC50 = 0.4 nM T61622 CCU45K 23625018 IC50 = 16 nM T61622 C7K8ED 23625020 IC50 = 2 nM T61622 CVM13T 23625022 IC50 = 2 nM T61622 C17ABC 23625024 IC50 = 7 nM T61622 CZ8J4Q 23625025 IC50 = 5 nM T61622 CEHO73 23625185 IC50 = 120 nM T61622 CYO5K8 23625483 IC50 = 0.8 nM T61622 CGX3T7 23625486 IC50 = 0.6 nM T61622 CB3HZ4 23625488 IC50 = 3 nM T61622 CX9CQ7 23625645 IC50 = 4 nM T61622 CNOF91 23625647 IC50 = 16 nM T61622 CNIR96 23625649 IC50 = 3 nM T61622 CO5S6B 23625789 IC50 = 4 nM T61622 CJ9U2T 23625790 IC50 = 95 nM T61622 C6YBA4 23625791 IC50 = 5 nM T61622 C5XB8Y 23625792 IC50 = 11 nM T61622 CA2YQ8 23625793 IC50 = 3 nM T61622 CMXJ30 23625795 IC50 = 0.6 nM T61622 CB46HG 23625796 IC50 = 1 nM T61622 C0Q1EO 23625798 IC50 = 1 nM T61622 C23CDF 23625951 IC50 = 4 nM T61622 CH8ED1 23625952 IC50 = 1 nM T61622 CDS2H1 23625953 IC50 = 6 nM T61622 C5ZP8A 23625954 IC50 = 19 nM T61622 C4SQ9L 23626112 IC50 = 2 nM T61622 CF6A8B 23626114 IC50 = 0.8 nM T61622 CXJ4Y7 23626116 IC50 = 18 nM T61622 CMG3X2 23626117 IC50 = 22 nM T61622 CXR5O6 23626119 IC50 = 2 nM T61622 CYH5O9 23626260 IC50 = 10 nM T61622 CRXC75 23626262 IC50 = 2 nM T61622 C4F5WP 23626264 IC50 = 10 nM T61622 CQB87W 23626266 IC50 = 12 nM T61622 CA24MD 23626267 IC50 = 10 nM T61622 C80GLA 23626268 IC50 = 1 nM T61622 C5U0IC 23626270 IC50 = 0.9 nM T61622 C8P3NG 23626272 IC50 = 3 nM T61622 CCJE50 23626274 IC50 = 4 nM T61622 CN26RU 23626276 IC50 = 0.8 nM T61622 CWOQ85 23626414 IC50 = 4 nM T61622 CC8QX0 23626416 IC50 = 1 nM T61622 CE8M1A 23626418 IC50 = 6 nM T61622 CR8KD6 23626420 IC50 = 1 nM T61622 CF5LW3 23626421 IC50 = 17 nM T61622 CTMD47 23626422 IC50 = 3 nM T61622 CPE12J 23626424 IC50 = 13 nM T61622 CN6T2C 23626426 IC50 = 2 nM T61622 CTB47R 23626428 IC50 = 1 nM T61622 CROK86 23626430 IC50 = 6 nM T61622 C8W5XY 23626573 IC50 = 1 nM T61622 C4NME7 23626575 IC50 = 3 nM T61622 CC9TY5 23626577 IC50 = 2 nM T61622 CBOG98 23626578 IC50 = 1 nM T61622 C0VC9Q 23626579 IC50 = 2 nM T61622 CIOZ62 23626580 IC50 = 1 nM T61622 CY4D2N 23626582 IC50 = 0.9 nM T61622 CBW34S 23626584 IC50 = 0.9 nM T61622 CG84BU 23626586 IC50 = 0.7 nM T61622 CP3KA6 23626588 IC50 = 1 nM T61622 CC65HN 23626745 IC50 = 0.3 nM T61622 C3Y9HD 23626746 IC50 = 16 nM T61622 CAB01E 23626748 IC50 = 7 nM T61622 CWG40S 23626749 IC50 = 2 nM T61622 CNHT35 23626750 IC50 = 1 nM T61622 C0YCP4 23626752 IC50 = 0.4 nM T61622 C4BYC8 23626754 IC50 = 0.6 nM T61622 C7EH6Q 23626756 IC50 = 3 nM T61622 C2V6QA 23626907 IC50 = 5 nM T61622 CMC58A 23626908 IC50 = 3 nM T61622 C3KQ2Y 23626909 IC50 = 2 nM T61622 CQDB27 23626913 IC50 = 2 nM T61622 C7HSL4 23628221 IC50 = 512 nM T61622 CYRO10 23628222 IC50 = 178 nM T61622 C9KA1C 23644725 IC50 = 4 nM T61622 C5L8SH 23644726 IC50 > 1000 nM T61622 CPB17O 23644727 IC50 = 0.68 nM T61622 C2Y3IA 23644728 IC50 = 340 nM T61622 CMP0N5 23647869 IC50 = 2700 nM T61622 C9QBH3 23647870 IC50 = 3900 nM T61622 CBXV89 23647871 IC50 = 235 nM T61622 C6AHK7 23647872 IC50 = 325 nM T61622 C34CZY 23647873 IC50 = 310 nM T61622 C0CZ1U 23647874 IC50 = 520 nM T61622 CN7DG0 23647875 IC50 = 132 nM T61622 CX1J7H 23647876 IC50 = 1040 nM T61622 CQ9JL3 23647877 IC50 = 430 nM T61622 CNY52R 23647878 IC50 = 220 nM T61622 CO0TZ5 23647879 IC50 = 206 nM T61622 CHDR91 23647880 IC50 = 325 nM T61622 C1SV6X 23647881 IC50 = 72 nM T61622 C1AQ9P 23647882 IC50 = 17 nM T61622 CTJ2P1 23647883 IC50 = 52 nM T61622 CU6E5F 23647884 IC50 = 245 nM T61622 C6NS9I 23647885 IC50 = 100 nM T61622 CD9IC3 23647886 IC50 = 1 nM T61622 CPX95O 23647887 IC50 = 175 nM T61622 CK9D8P 23647888 IC50 = 66 nM T61622 CX50BA 23647889 IC50 = 60 nM T61622 C37JMS 23647890 IC50 > 40 nM T61622 CU6D5S 23647891 IC50 = 7 nM T61622 CJ97BQ 23647892 IC50 = 7 nM T61622 CXP2G5 23647893 IC50 = 0.8 nM T61622 C3JBX4 23647894 IC50 = 860 nM T61622 C71DGY 23647895 IC50 = 890 nM T61622 C03JFU 23647896 IC50 = 1080 nM T61622 C5LU8P 23647897 IC50 = 43 nM T61622 C2YVQ3 23647898 IC50 = 3 nM T61622 C4H5PR 23647899 IC50 = 6 nM T61622 CW6Y9I 23647900 IC50 = 200 nM T61622 CMF8R6 23647901 IC50 = 630 nM T61622 CR7CO9 23647902 IC50 = 2 nM T61622 CX37CO 23647903 IC50 = 62 nM T61622 CMG8T2 23647904 IC50 = 182 nM T61622 C9H7NY 23647905 IC50 = 41 nM T61622 CHA50G 23647906 IC50 = 188 nM T61622 C3MSV0 23647907 IC50 = 48 nM T61622 C2Z0KQ 23647908 IC50 = 198 nM T61622 CD8XH5 23647909 IC50 = 120 nM T61622 CF9EK5 23647910 IC50 = 91 nM T61622 CB1PL5 23647911 IC50 = 606 nM T61622 CQ9I4F 23647912 IC50 = 550 nM T61622 C9H0EC 23647913 IC50 = 450 nM T61622 CN61YJ 23647914 IC50 = 1200 nM T61622 CL56AY 23647915 IC50 = 58 nM T61622 C8PXO6 23726071 IC50 = 1 nM T61622 C1AYW2 24742297 IC50 = 0.17 nM T61622 CC0X4Z 24742462 IC50 = 0.17 nM T61622 C80ACG 24742640 IC50 = 0.28 nM T61622 C7W3NH 24742904 IC50 = 0.12 nM T61622 CF90TW 24742991 IC50 = 0.44 nM T61622 C1BO9N 24743241 IC50 = 0.5 nM T61622 CO6S0Y 24744682 IC50 = 0.24 nM T61622 CS3M2E 24744683 IC50 = 0.15 nM T61622 CK84DL 24836809 IC50 = 0.8 nM T61622 CA15QU 24864107 IC50 = 0.2 nM T61622 C8OG1C 24875446 IC50 = 3 nM T61622 CZEK21 24875911 IC50 = 1 nM T61622 CR7PH1 24876739 IC50 = 3 nM T61622 CG0Z5M 24883482 IC50 > 250000 nM T61622 CY08DL 24883483 IC50 > 250000 nM T61622 C32SYP 24950594 IC50 = 2040 nM T61622 CCO20I 24953169 IC50 = 0.028 nM T61622 CC0U6X 24953170 IC50 = 0.097 nM T61622 CO41IK 24953519 IC50 = 0.046 nM T61622 CER42Y 24966529 IC50 = 2 nM T61622 CMN4L1 24966889 IC50 = 1 nM T61622 C2A9HN 24966890 IC50 = 1.1 nM T61622 CQR20U 24968904 IC50 = 1 nM T61622 CO7MQ2 25069561 IC50 = 30100 nM T61622 C8ANG7 25070193 IC50 = 6000 nM T61622 CM37LQ 25072736 IC50 = 8600 nM T61622 C0UO6V 25073049 IC50 = 16900 nM T61622 CRK8L4 25077620 Ki = 2000 nM T61622 C2UWA1 25096462 Ki = 21 nM T61622 CG6H9T 25099190 IC50 = 0.67 nM T61622 CXBZ57 25118294 IC50 = 9 nM T61622 CJM41E 25119356 IC50 = 23.4 nM T61622 C8HI9Y 25119357 IC50 = 12.4 nM T61622 CGL63Q 25119716 IC50 = 0.03 nM T61622 CQ8Y7T 25120419 IC50 = 0.04 nM T61622 CXL3Q8 25121114 IC50 = 0.06 nM T61622 C2S1LG 25121469 IC50 = 0.01 nM T61622 C1RBQ7 25122183 IC50 = 0.027 nM T61622 CYWO57 25122184 IC50 = 0.064 nM T61622 CNTF43 25127621 IC50 = 7700 nM T61622 C4E0MJ 25127622 IC50 = 4800 nM T61622 CWF5Z3 25143506 IC50 = 0.2 nM T61622 CF5H0Z 25191496 IC50 = 6 nM T61622 CY3W1J 25191615 IC50 = 19.7 nM T61622 CB4G1Z 25191616 IC50 = 0.44 nM T61622 C5WUF9 25191617 IC50 = 7.41 nM T61622 CDB8V6 25191618 IC50 = 1.7 nM T61622 CX9VC3 25191619 IC50 = 44.4 nM T61622 CIY0K8 25191742 IC50 = 1151 nM T61622 CS6ET2 25191743 IC50 = 47.6 nM T61622 CNGA86 25191744 IC50 = 0.09 nM T61622 C58INK 25191745 IC50 = 0.52 nM T61622 C1DQU8 25242438 IC50 = 0.38 nM T61622 CIH75Y 42615261 IC50 = 0.47 nM T61622 COUG86 42627773 IC50 = 88 nM T61622 C9PL8Z 42641334 IC50 = 318 nM T61622 C2ICV4 42641452 IC50 = 62 nM T61622 C6MX0U 42641453 IC50 = 6.4 nM T61622 CV7U9F 42641563 IC50 = 23 nM T61622 CMI2E8 42641564 IC50 = 54 nM T61622 CSK0M9 42641566 IC50 = 120 nM T61622 CQIV32 42641674 IC50 = 139 nM T61622 CA5TW1 42641905 IC50 = 1.2 nM T61622 CQS4U7 42642010 IC50 = 1.2 nM T61622 CIX54O 42642011 IC50 = 1.1 nM T61622 CH6V4W 44143374 IC50 = 308 nM T61622 CVT0R7 44143375 IC50 = 55 nM T61622 CN5G1Q 44143376 IC50 = 5.5 nM T61622 C02MOI 44143377 IC50 = 764 nM T61622 C8YB9A 44143378 IC50 = 58 nM T61622 CEC01K 44143379 IC50 = 39 nM T61622 CNUE94 44143380 IC50 = 609 nM T61622 C6HO8P 44143381 IC50 = 40 nM T61622 C0HN3L 44143382 IC50 = 4 nM T61622 C6DFG5 44143383 IC50 = 11 nM T61622 CA2TF5 44143384 IC50 = 125 nM T61622 C7F0ZK 44143385 IC50 = 490 nM T61622 C0NP5H 44143386 IC50 = 21 nM T61622 CEH6N1 44143387 IC50 = 21 nM T61622 CW01UO 44143388 IC50 = 7 nM T61622 C3OP8W 44143389 IC50 = 16 nM T61622 CY60MQ 44143390 IC50 = 7 nM T61622 C1WY7J 44143391 IC50 = 4 nM T61622 CDYB08 44143392 IC50 = 2.5 nM T61622 CYLG05 44143393 IC50 = 9 nM T61622 C6N2MR 44143394 IC50 = 13 nM T61622 C23TCK 44143395 IC50 = 47 nM T61622 C89UPC 44143396 IC50 = 0.13 nM T61622 C2Y7LU 44143397 IC50 = 37 nM T61622 CUH37T 44143398 IC50 = 389 nM T61622 CBG10Y 44143399 IC50 = 69 nM T61622 C0X6FT 44143400 IC50 = 6 nM T61622 CV0E5Z 44143401 IC50 = 46 nM T61622 CTPM47 44143402 IC50 = 0.14 nM T61622 CB0JW1 44143403 IC50 = 0.1 nM T61622 CF94RU 44143404 IC50 = 3.5 nM T61622 C3RX9S 44143405 IC50 = 0.9 nM T61622 C26BAU 44157990 IC50 = 6.8 nM T61622 CGIH90 44157991 IC50 = 8.3 nM T61622 CAI71N 44157992 IC50 = 25 nM T61622 CTIX02 44158056 IC50 = 5.2 nM T61622 C0UP1R 44158057 IC50 = 0.62 nM T61622 C12RWX 44158060 IC50 = 130 nM T61622 CC3Z6V 44158061 IC50 = 4.8 nM T61622 C7R9JN 44158062 IC50 = 1.6 nM T61622 C1N7DE 44158063 IC50 = 3.2 nM T61622 CWR4T6 44158064 IC50 = 7.7 nM T61622 C68ABV 44158065 IC50 = 1.4 nM T61622 CDMV70 44158066 IC50 = 38 nM T61622 CHG2J9 44158067 IC50 = 19 nM T61622 C37ILS 44158119 IC50 = 16 nM T61622 C6UL1E 44158120 IC50 = 2.4 nM T61622 C8S3DK 44158121 IC50 = 5.2 nM T61622 CW7P1M 44158124 IC50 = 7500 nM T61622 C4JWY5 44158125 IC50 = 0.83 nM T61622 CKPF81 44158126 IC50 = 0.29 nM T61622 CKJ0I7 44158127 IC50 = 8.5 nM T61622 CN2CM6 44158128 IC50 = 1100 nM T61622 CVAH76 44158191 IC50 = 257 nM T61622 C96OBG 44158192 IC50 = 0.28 nM T61622 C1EZ4W 44158193 IC50 = 4.9 nM T61622 CIX23Z 44158194 IC50 = 7 nM T61622 C4QKI9 44158195 IC50 = 116 nM T61622 C5T7DZ 44158196 IC50 = 640 nM T61622 CC1W2Z 44158197 IC50 = 1.5 nM T61622 CZKO30 44158198 IC50 = 0.25 nM T61622 CKX6G7 44158199 IC50 = 415 nM T61622 CUH7J8 44158200 IC50 = 29 nM T61622 C73RDZ 44158201 IC50 = 1.5 nM T61622 C8ZU0W 44158202 IC50 = 0.3 nM T61622 C0BLJ5 44158272 IC50 = 4.6 nM T61622 CXGK65 44158273 IC50 = 54 nM T61622 CFB76L 44158274 IC50 = 0.33 nM T61622 C2M6EW 44158276 IC50 = 0.2 nM T61622 C4SM7F 44158277 IC50 = 1.4 nM T61622 CI21LT 44158432 IC50 = 3160 nM T61622 C8GZU4 44158434 IC50 = 3410 nM T61622 CYI40G 44158435 IC50 = 420 nM T61622 CI3A5C 44158647 IC50 = 18 nM T61622 C97YHS 44158650 IC50 = 9 nM T61622 C1N2FV 44158681 IC50 = 250 nM T61622 CD9M3Y 44158682 IC50 = 939 nM T61622 CZ41WH 44158683 IC50 = 120 nM T61622 CFZ6R9 44158791 IC50 = 12 nM T61622 COC9R6 44158792 IC50 = 24 nM T61622 C7X8LD 44158793 IC50 = 57 nM T61622 CX71KW 44158794 IC50 = 74 nM T61622 CO1Y5T 44158795 IC50 = 590 nM T61622 CV2MD3 44158796 IC50 = 1600 nM T61622 CP1LF7 44158906 IC50 = 123 nM T61622 C1L7QO 44158907 IC50 = 3400 nM T61622 C1PTY2 44158908 IC50 = 520 nM T61622 C5Z1EJ 44158909 IC50 = 100 nM T61622 CH7NU2 44158910 IC50 = 200 nM T61622 C1Q8LJ 44159019 IC50 = 494 nM T61622 COX7S6 44159020 IC50 = 761 nM T61622 C69KBX 44159021 IC50 = 14 nM T61622 CUEK39 44159022 IC50 = 27 nM T61622 C3P9BN 44160196 IC50 = 5 nM T61622 CTC3U2 44160197 IC50 = 21 nM T61622 CPQ9X1 44194118 IC50 = 2 nM T61622 CVS7E4 44195154 IC50 = 2 nM T61622 C1F0ZO 44213183 IC50 = 0.8 nM T61622 CZ85SD 44236883 IC50 > 250000 nM T61622 CCJN58 44236884 IC50 > 250000 nM T61622 CZIF43 44236885 IC50 > 250000 nM T61622 CC83SD 44236886 IC50 > 250000 nM T61622 C85DAM 44236887 IC50 > 250000 nM T61622 C15SQV 44236888 IC50 > 250000 nM T61622 CNB0E9 44236889 Ki = 5700 nM T61622 C6DR4L 44236890 IC50 > 250000 nM T61622 C6N2KH 44236891 Ki = 16000 nM T61622 C1JTG2 44244046 IC50 > 1991000 nM T61622 CX7G6U 44265557 IC50 = 5 nM T61622 CC48GO 44265653 IC50 = 0.23 nM T61622 CW87GY 44267805 IC50 = 20000 nM T61622 CEU04K 44267824 IC50 = 1200000 nM T61622 C9ZKP6 44267838 IC50 = 80000 nM T61622 C4XY0A 44274653 IC50 = 580 nM T61622 CJ1AB3 44274654 IC50 = 200000 nM T61622 CPB4S0 44276584 IC50 = 20 nM T61622 C2XDH5 44276585 IC50 = 3.6 nM T61622 CJKL06 44276634 IC50 = 6 nM T61622 CT06ND 44276669 IC50 = 5.2 nM T61622 CC6S5N 44276707 Ki = 146000 nM T61622 C4Z6LQ 44276708 Ki = 80000 nM T61622 C7C4IB 44276829 Ki = 1000000 nM T61622 CDE60K 44276843 Ki = 400000 nM T61622 C0EJN4 44278004 IC50 = 4 nM T61622 C0H5GJ 44278005 IC50 = 0.7 nM T61622 CZPF67 44278006 IC50 = 2.4 nM T61622 CW8MU1 44278055 IC50 = 0.4 nM T61622 CE4GP7 44278067 IC50 = 7.5 nM T61622 C7CTW5 44278182 IC50 = 2 nM T61622 CW2HI5 44278242 IC50 = 0.55 nM T61622 C6H8NU 44278243 IC50 = 55 nM T61622 C4KD1W 44278281 IC50 = 4.8 nM T61622 C52XKV 44278282 IC50 = 26 nM T61622 CHU97J 44278306 IC50 = 5.4 nM T61622 CQLD70 44278337 IC50 = 20 nM T61622 CP2V8F 44278393 IC50 = 10000 nM T61622 CY5G4Q 44278465 IC50 = 370 nM T61622 CHO3F4 44278466 IC50 = 10 nM T61622 CGK61B 44278482 Ki = 1000 nM T61622 CA9ER5 44278603 IC50 = 164 nM T61622 C0L1XB 44278672 IC50 = 2 nM T61622 CUM3W7 44278696 IC50 = 0.32 nM T61622 C0PGY3 44278697 IC50 = 0.21 nM T61622 CP2IC9 44278742 IC50 = 0.87 nM T61622 CB6Z8Q 44278754 IC50 = 0.44 nM T61622 CV5Z2K 44278755 IC50 = 12.3 nM T61622 CZ3JV0 44278756 IC50 = 0.69 nM T61622 CL86BE 44278763 IC50 = 2.96 nM T61622 CB9X3R 44278764 IC50 = 0.24 nM T61622 C20IBP 44278779 IC50 = 2.33 nM T61622 C8CJ5U 44278793 IC50 = 10 nM T61622 CR0U9J 44278822 IC50 = 0.46 nM T61622 C97YGC 44278880 IC50 = 0.7 nM T61622 CQZU21 44278890 IC50 = 0.81 nM T61622 C83MJY 44278917 IC50 = 0.62 nM T61622 CD2LZ6 44278918 IC50 = 0.22 nM T61622 C1HG4D 44278937 IC50 = 1.89 nM T61622 C15FIE 44278947 IC50 = 740 nM T61622 CV6JM2 44278948 IC50 > 1000000 nM T61622 CTSR15 44278950 IC50 = 87 nM T61622 CCR49J 44278956 IC50 = 97.8 nM T61622 C3F7YI 44278960 IC50 = 160 nM T61622 CO6H8B 44278968 IC50 = 55 nM T61622 C01THG 44278974 IC50 = 1.5 nM T61622 C19UFM 44278975 IC50 = 0.79 nM T61622 COT30Q 44278979 IC50 = 53 nM T61622 C9S6CA 44278994 IC50 = 22 nM T61622 C5PFN2 44278995 IC50 = 0.4 nM T61622 C3T0IN 44279009 IC50 = 1.5 nM T61622 C0AK8S 44279012 IC50 = 1.49 nM T61622 CM9A4R 44279024 IC50 = 100 nM T61622 CM7C8F 44279044 IC50 = 19.1 nM T61622 CGZ5J4 44279045 IC50 = 0.42 nM T61622 CWS85T 44279062 IC50 = 0.57 nM T61622 CD9C6F 44279063 IC50 = 0.28 nM T61622 CFAM56 44279154 IC50 = 540 nM T61622 CT39ZH 44279174 IC50 = 8 nM T61622 C6W7NQ 44279189 IC50 = 40000 nM T61622 C2GQT7 44279226 IC50 = 210 nM T61622 C0PCN7 44279227 IC50 = 25000 nM T61622 C47JNO 44279247 IC50 = 1200000 nM T61622 CZ4E0Y 44279250 IC50 = 10000 nM T61622 CMN4X8 44279264 IC50 = 3.3 nM T61622 CSM9W8 44279283 IC50 = 6.4 nM T61622 CIQ60W 44279315 IC50 = 160 nM T61622 CE4R7K 44279318 IC50 = 810 nM T61622 C50NBC 44279451 IC50 = 91 nM T61622 C74ZHL 44279486 IC50 = 41 nM T61622 C78QLB 44279501 IC50 = 880 nM T61622 CN5QM2 44279522 IC50 = 160 nM T61622 C2MYI8 44279529 IC50 = 820 nM T61622 CA6NL0 44279530 IC50 = 590 nM T61622 CA9TF2 44279541 IC50 = 2600 nM T61622 CY1M6D 44279543 IC50 = 580 nM T61622 CJX7T6 44279544 IC50 = 26 nM T61622 CH7E2Q 44279557 IC50 = 4 nM T61622 CV5NC3 44279658 IC50 = 2.3 nM T61622 CDS68G 44279659 IC50 = 190 nM T61622 CB7CS0 44279694 IC50 = 380 nM T61622 CLH09N 44279745 IC50 = 220 nM T61622 C9R0JK 44279813 IC50 = 0.79 nM T61622 CT48DZ 44279814 IC50 = 0.38 nM T61622 C8PEH9 44279815 IC50 = 0.77 nM T61622 CPNL53 44279834 IC50 = 1.4 nM T61622 C3ROG8 44279835 IC50 = 0.7 nM T61622 CKVU23 44279850 IC50 = 33 nM T61622 C6N9OR 44279924 IC50 = 0.48 nM T61622 CP9X2R 44279925 IC50 = 0.63 nM T61622 C1MYQ7 44279926 IC50 = 1.4 nM T61622 CV17XK 44279952 IC50 = 4.4 nM T61622 CMQ6L0 44279953 IC50 = 1.9 nM T61622 CKEG34 44279959 IC50 = 0.63 nM T61622 CI52NR 44279972 IC50 = 23 nM T61622 C9W6XD 44279973 IC50 = 0.59 nM T61622 CZ9LF3 44279989 IC50 = 14 nM T61622 CU58TM 44279990 IC50 = 7 nM T61622 C4Y3MI 44280015 IC50 = 1.2 nM T61622 CUDB58 44280040 IC50 = 27 nM T61622 CZ59XK 44280057 IC50 = 15 nM T61622 C9ZE8N 44280358 IC50 = 0.37 nM T61622 CL3PA2 44282469 Ki = 1180000 nM T61622 C64CPN 44286912 IC50 = 1.7 nM T61622 C3I5YC 44286933 IC50 = 1.8 nM T61622 C7FBO9 44286934 IC50 = 38 nM T61622 CA9R2O 44286998 IC50 = 1.4 nM T61622 CUO12K 44287040 IC50 = 1.9 nM T61622 C09XSI 44287041 IC50 = 1.6 nM T61622 C9OH8C 44287042 IC50 = 1.7 nM T61622 C0KEY5 44287424 IC50 = 700 nM T61622 CW8FP3 44287425 IC50 = 3700 nM T61622 CQ5I3G 44287451 IC50 > 100000 nM T61622 C8YDA7 44287452 IC50 = 32000 nM T61622 CX5K9Q 44287613 IC50 = 1.2 nM T61622 CT51WO 44287641 IC50 = 4300 nM T61622 CRQ3C2 44287642 IC50 = 13000 nM T61622 C2AO9R 44287674 IC50 = 2900 nM T61622 C6U5NA 44287804 IC50 = 58000 nM T61622 C5CL0E 44287870 IC50 = 79000 nM T61622 C1I6HF 44287871 IC50 = 10000 nM T61622 CBFZ73 44287872 IC50 = 2700 nM T61622 CYX58N 44287873 IC50 = 2100 nM T61622 CCT87P 44289279 Ki = 4.8 nM T61622 CE17WQ 44289280 Ki = 154 nM T61622 CBX4L9 44290111 IC50 = 70 nM T61622 CA89WZ 44290137 IC50 = 2000 nM T61622 C6WZQ7 44290138 IC50 > 30000 nM T61622 CC50RT 44290139 IC50 = 600 nM T61622 CEW26C 44290197 IC50 = 6000 nM T61622 CQZ47C 44290291 IC50 > 30000 nM T61622 C89GCV 44290303 IC50 = 6400 nM T61622 CA6BD3 44290304 IC50 > 30000 nM T61622 CH9V0N 44290305 IC50 > 30000 nM T61622 CT98LQ 44290313 IC50 = 40 nM T61622 C9XIA6 44290367 IC50 = 800 nM T61622 CI5LH7 44290381 IC50 = 900 nM T61622 C65IBX 44290442 IC50 > 30000 nM T61622 C53NQS 44290443 IC50 = 5000 nM T61622 C1P8MU 44290466 IC50 > 30000 nM T61622 CE9J6W 44290467 IC50 > 30000 nM T61622 CBD6A4 44291251 IC50 = 15 nM T61622 CI9X2M 44291252 IC50 = 0.5 nM T61622 CIW20X 44291312 IC50 = 3.2 nM T61622 CFRX32 44291388 IC50 = 14 nM T61622 C2D0FM 44292177 IC50 = 37000 nM T61622 CXI3Q8 44292210 IC50 > 100000 nM T61622 CV3RH4 44292211 IC50 > 100000 nM T61622 CXAN93 44292758 IC50 = 10 nM T61622 C1AU3D 44292774 IC50 = 120 nM T61622 CTX04Y 44292788 IC50 = 44 nM T61622 CP7I3F 44292789 IC50 = 200 nM T61622 CWZG41 44293026 IC50 = 1.1 nM T61622 CX8C3H 44293440 IC50 = 3.3 nM T61622 CA8XD3 44293742 IC50 = 0.9 nM T61622 C4M6AO 44293992 IC50 = 5.1 nM T61622 CH2O9I 44294053 IC50 = 1.4 nM T61622 C6I8UF 44297360 IC50 = 4 nM T61622 CW29IT 44297438 IC50 = 20 nM T61622 CIM7K8 44297439 IC50 = 20 nM T61622 CW6SL9 44297444 IC50 = 4 nM T61622 C68ZGW 44297445 IC50 = 20 nM T61622 C8VBX1 44297462 IC50 = 0.4 nM T61622 C1OVP3 44297499 IC50 = 7 nM T61622 CQW87S 44297500 IC50 = 2800 nM T61622 C4FPR3 44297524 IC50 = 340 nM T61622 C86JOX 44297527 IC50 = 15 nM T61622 C09DVE 44297615 IC50 = 15 nM T61622 CKI6T3 44297620 IC50 = 6 nM T61622 CI1WM0 44297621 IC50 = 2 nM T61622 C2M4LC 44297662 IC50 = 12 nM T61622 CLFY29 44297663 IC50 = 330 nM T61622 C5IJ0V 44297664 IC50 = 480 nM T61622 C3CNO6 44297670 IC50 = 730 nM T61622 CIEX86 44297827 IC50 = 6.7 nM T61622 C3M6DF 44297942 Ki = 36 nM T61622 C0U3GF 44297957 Ki = 50 nM T61622 C5B7MZ 44297958 Ki = 0.12 nM T61622 CN1GV3 44297959 Ki = 0.98 nM T61622 C2BZP8 44297960 Ki = 20 nM T61622 CY1RJ3 44297968 Ki = 0.04 nM T61622 CT94RA 44298033 Ki = 36 nM T61622 C7RPE2 44298059 Ki = 120 nM T61622 C0Z8EC 44298072 Ki = 6 nM T61622 C84GDY 44298379 IC50 = 8200 nM T61622 CH2CA9 44298391 IC50 = 880 nM T61622 CZ71MH 44298408 IC50 = 340 nM T61622 C81TZJ 44298422 IC50 = 260 nM T61622 CF06RO 44298423 IC50 = 800 nM T61622 CBDI95 44298435 IC50 = 600 nM T61622 C3JU6B 44298437 IC50 = 48 nM T61622 CQ06FJ 44298461 IC50 = 13 nM T61622 CJ2X6U 44298499 IC50 = 3000 nM T61622 C0EM3C 44298518 IC50 = 140 nM T61622 CXEH24 44298519 IC50 = 790 nM T61622 CJ2TS7 44298520 IC50 = 420 nM T61622 CVXR31 44300316 IC50 = 3.3 nM T61622 C1SZ3V 44300327 IC50 = 1.4 nM T61622 CTW7Y5 44300345 IC50 = 92 nM T61622 CJ6U4L 44300358 IC50 = 20 nM T61622 CW6SO1 44300359 IC50 = 280 nM T61622 C5BTY6 44300360 IC50 = 170 nM T61622 CP3BY8 44300380 IC50 = 0.59 nM T61622 CD5P7L 44300403 IC50 = 54 nM T61622 C9QS1D 44300409 IC50 = 64 nM T61622 CGE48Q 44300410 IC50 = 6.8 nM T61622 C3HY5E 44300411 IC50 = 880 nM T61622 CCK15B 44300412 IC50 = 50 nM T61622 C63NWS 44300416 IC50 = 140 nM T61622 CBT5H1 44300430 IC50 = 0.99 nM T61622 CMDF96 44300431 IC50 = 940 nM T61622 C2D9WM 44300457 IC50 = 120 nM T61622 CKI78D 44300491 IC50 = 9 nM T61622 C74SCJ 44300917 IC50 = 1.4 nM T61622 C5YEK2 44300918 IC50 = 0.68 nM T61622 C07UBA 44300955 IC50 = 0.19 nM T61622 C18WEQ 44300956 IC50 = 27 nM T61622 CTMD90 44300959 IC50 = 0.18 nM T61622 C2Q5ZD 44301266 IC50 = 15 nM T61622 C81WME 44301267 IC50 = 0.95 nM T61622 CA2GS3 44301665 IC50 = 0.23 nM T61622 CGH3U9 44301873 IC50 = 2.7 nM T61622 C2G6YV 44301892 IC50 = 1.7 nM T61622 C3ORT1 44301893 IC50 = 1.7 nM T61622 CD1YK3 44301912 IC50 = 3.4 nM T61622 C1WLN8 44301941 IC50 = 46 nM T61622 C4D2WJ 44301961 IC50 = 27 nM T61622 C8OBV6 44301962 IC50 = 0.49 nM T61622 C9B0VW 44301974 IC50 = 6.9 nM T61622 C6WPL8 44301975 IC50 = 0.59 nM T61622 CLF1G8 44301976 IC50 = 7.3 nM T61622 CX79EY 44301978 IC50 = 12 nM T61622 CJT20G 44302154 IC50 = 26 nM T61622 C5GD2C 44302155 IC50 = 100 nM T61622 CSU08N 44303448 IC50 = 0.2 nM T61622 C24HAR 44303449 IC50 = 190 nM T61622 CNOC05 44303450 IC50 = 190 nM T61622 CLQ6J5 44303672 IC50 = 32 nM T61622 CVF6Y2 44303747 IC50 = 25 nM T61622 C5M4ZK 44303748 IC50 = 1400 nM T61622 CDMI23 44303772 IC50 = 60 nM T61622 CSF79G 44303773 IC50 = 5.8 nM T61622 C96AKM 44303994 IC50 = 3.6 nM T61622 CC1BQ9 44303995 IC50 = 0.42 nM T61622 CCZ2I3 44304033 IC50 = 101 nM T61622 C3L4PI 44304145 IC50 = 325 nM T61622 CBTJ72 44304146 IC50 = 146 nM T61622 CUB84O 44304257 IC50 = 11.5 nM T61622 C15RPV 44304333 IC50 = 373 nM T61622 CT1N0I 44305053 IC50 = 0.35 nM T61622 CW71IO 44306396 IC50 = 120 nM T61622 CCOH58 44307374 Ki = 0.051 nM T61622 CCPJ83 44308283 IC50 = 430 nM T61622 CZ02PM 44308293 IC50 = 70 nM T61622 CEO5N1 44308356 IC50 = 25 nM T61622 C9JAL0 44308357 IC50 = 40 nM T61622 C7SHK5 44308358 IC50 = 20 nM T61622 CMBL48 44308399 IC50 = 150 nM T61622 CHL3O7 44314473 IC50 > 100000 nM T61622 CPEF43 44314483 IC50 = 330 nM T61622 C1JGY2 44314484 IC50 = 1.6 nM T61622 C0XUE2 44314485 IC50 = 3.7 nM T61622 CFWK98 44314488 IC50 = 1.9 nM T61622 CH9I7M 44314498 IC50 = 48 nM T61622 CPQ56L 44314499 IC50 = 6.8 nM T61622 CS67LQ 44314500 IC50 = 1.7 nM T61622 CP30DX 44314501 IC50 = 1 nM T61622 C9NJY3 44314576 IC50 = 32000 nM T61622 CEW8T9 44314869 IC50 = 63 nM T61622 CH9PX2 44314870 IC50 = 290 nM T61622 CF9K7N 44314903 IC50 = 1920 nM T61622 C6FOV3 44315276 IC50 = 26 nM T61622 C0CQ9A 44317192 Ki = 800 nM T61622 CQ5F2W 44317193 Ki = 2500 nM T61622 CG5PQ0 44319473 IC50 = 870 nM T61622 CZ8L3U 44319490 IC50 = 31000 nM T61622 CK0Z8O 44319812 IC50 = 710 nM T61622 CAYK67 44319816 IC50 = 40000 nM T61622 CJN83A 44319822 IC50 = 1900 nM T61622 CCPY04 44319823 IC50 = 520 nM T61622 CHX49L 44319865 IC50 = 130 nM T61622 COJ6R0 44319879 IC50 = 860 nM T61622 C0MAW3 44319911 IC50 = 2300 nM T61622 C8N1OQ 44319983 IC50 = 63 nM T61622 C1VUC3 44319985 IC50 = 430 nM T61622 C2NM3D 44320020 IC50 = 3.4 nM T61622 CX3IT1 44320039 IC50 = 880 nM T61622 C7G9LV 44320059 IC50 = 0.91 nM T61622 C1LJW7 44320156 IC50 = 0.48 nM T61622 C8TE2K 44320162 IC50 = 0.35 nM T61622 CUF79D 44320175 IC50 = 4.1 nM T61622 CR2NI0 44320182 IC50 = 750 nM T61622 CX39TP 44320278 IC50 = 1400 nM T61622 C4KPI3 44320299 IC50 = 2740 nM T61622 CIE9T8 44320330 IC50 = 33 nM T61622 CNJ53Z 44320331 IC50 = 2.34 nM T61622 CIU5D2 44320332 IC50 = 26 nM T61622 CVO4Z1 44320333 IC50 = 1500 nM T61622 CI30HL 44320334 IC50 = 240 nM T61622 C1GEZ5 44320563 IC50 = 13.7 nM T61622 CR2T3Y 44320564 IC50 = 0.16 nM T61622 C9FIC2 44320565 IC50 = 0.581 nM T61622 C32TRA 44320597 IC50 = 0.27 nM T61622 CS7XD5 44321765 IC50 = 0.3 nM T61622 C2OFK8 44321766 IC50 = 0.2 nM T61622 CZ45LH 44322035 IC50 = 0.3 nM T61622 CQ09YG 44322074 IC50 = 0.9 nM T61622 C3N9LQ 44322075 IC50 = 13 nM T61622 CK0BQ2 44322083 IC50 = 44 nM T61622 CNT69K 44322084 IC50 = 0.2 nM T61622 CN58AQ 44322086 IC50 > 1 nM T61622 C1G0FY 44322087 IC50 = 0.6 nM T61622 C9VU8M 44322106 IC50 = 1600 nM T61622 C4UA0T 44322122 IC50 = 1100 nM T61622 CDJ1K8 44322317 IC50 = 0.3 nM T61622 CA0NB2 44322329 IC50 = 16000 nM T61622 C84IWM 44322382 IC50 = 1200 nM T61622 C07LPV 44322383 IC50 = 110 nM T61622 CVX76B 44322416 IC50 = 5100 nM T61622 C6TKY0 44324268 IC50 = 610 nM T61622 CX07YM 44324673 IC50 = 6.2 nM T61622 CN40SK 44324715 IC50 = 110 nM T61622 C4BCA9 44324785 IC50 = 1.9 nM T61622 C1U4PE 44324786 IC50 = 10 nM T61622 C7AWV1 44324787 IC50 = 1000 nM T61622 C8RE6I 44324788 IC50 = 7000 nM T61622 C9RS5I 44324881 IC50 = 470000 nM T61622 C98DMN 44324882 IC50 > 1000000 nM T61622 CXO6E2 44324883 IC50 = 14000 nM T61622 CWO54M 44325065 IC50 = 1.5 nM T61622 C40VEC 44325066 IC50 = 0.7 nM T61622 CQKG14 44325067 IC50 = 0.6 nM T61622 C8U9OP 44325109 IC50 = 0.35 nM T61622 CP2F5Y 44325110 IC50 = 11 nM T61622 CTGO85 44325120 IC50 = 21000 nM T61622 CVM9L8 44325121 IC50 = 64 nM T61622 CNT9X5 44325127 IC50 > 1000000 nM T61622 C6WN8A 44325167 IC50 > 1000000 nM T61622 C58FRI 44325168 IC50 = 310000 nM T61622 CS4O2Q 44325178 IC50 = 1.7 nM T61622 CG93FX 44325179 IC50 = 52000 nM T61622 C5SWD8 44325306 IC50 > 1000000 nM T61622 C1SOQ5 44325307 IC50 > 1000000 nM T61622 CD4PL7 44325308 IC50 > 1000000 nM T61622 C5OG8T 44325314 IC50 > 1000000 nM T61622 CE8ID3 44325315 IC50 = 680000 nM T61622 CMO79N 44325330 IC50 > 1000000 nM T61622 CCFB46 44325334 IC50 = 1500 nM T61622 COZ76T 44325336 IC50 = 14000 nM T61622 CBS26Y 44325350 IC50 = 240 nM T61622 C9Q8VI 44325369 IC50 = 39000 nM T61622 C27MNR 44325380 IC50 = 4000 nM T61622 CJS2D1 44325393 IC50 = 3000 nM T61622 COP31S 44325394 IC50 = 2000 nM T61622 CK56IJ 44325434 IC50 = 290 nM T61622 C98LYK 44325449 IC50 = 140000 nM T61622 C45CKG 44325450 IC50 = 240 nM T61622 CCQS25 44325466 IC50 > 1000000 nM T61622 C2K1MR 44325481 IC50 > 1000000 nM T61622 CU56KN 44325499 IC50 = 3500 nM T61622 CM6S5B 44326549 IC50 = 7.2 nM T61622 CST6G9 44326648 IC50 = 73 nM T61622 CAHZ92 44327253 IC50 = 0.25 nM T61622 C1M0ZQ 44327266 IC50 = 0.31 nM T61622 C37CUD 44327267 IC50 = 0.14 nM T61622 C05XEG 44327278 IC50 = 0.54 nM T61622 C4ME7H 44327315 IC50 = 0.69 nM T61622 CU83SP 44327316 IC50 = 1.1 nM T61622 CMZE09 44327317 IC50 = 4.2 nM T61622 CXS26D 44327449 IC50 = 0.47 nM T61622 CVA9J6 44327639 IC50 = 0.17 nM T61622 CCRT26 44331132 IC50 = 280 nM T61622 C93IQG 44331133 IC50 = 1400 nM T61622 C4LZ2Q 44331134 IC50 = 1200 nM T61622 C1V7JY 44331135 IC50 > 100000 nM T61622 CJX17Q 44331167 IC50 = 2700 nM T61622 CXZ84U 44331168 IC50 = 4600 nM T61622 C06RHF 44331191 IC50 = 69000 nM T61622 CAD7O0 44332761 IC50 = 1 nM T61622 CU1RS5 44332762 IC50 = 16 nM T61622 CPG31N 44332763 IC50 = 1.6 nM T61622 C6RQ9P 44332769 IC50 = 2100 nM T61622 CR08NU 44332784 IC50 = 5000 nM T61622 C3IL7O 44332786 IC50 = 0.38 nM T61622 CBUA51 44332787 IC50 = 8300 nM T61622 C7Y1BU 44332789 IC50 > 100000 nM T61622 CW5PV2 44332790 IC50 = 5800 nM T61622 CPF4T1 44332791 IC50 = 1300 nM T61622 C2XL8O 44332792 IC50 = 14 nM T61622 CNC76P 44332794 IC50 = 370000 nM T61622 CJ82NK 44332795 IC50 = 6.8 nM T61622 CZ51KB 44332796 IC50 = 21 nM T61622 C1RI2X 44332797 IC50 = 0.53 nM T61622 CK9GF3 44332798 IC50 = 3.8 nM T61622 C54DNZ 44332799 IC50 = 31 nM T61622 CLU0C6 44332800 IC50 = 0.1 nM T61622 C79CMX 44332881 IC50 ~ 100000 nM T61622 C86EJX 44332882 IC50 = 200 nM T61622 C6CIX7 44332883 IC50 = 0.31 nM T61622 CPF13H 44335353 IC50 > 10000 nM T61622 C19UEW 44339873 IC50 = 4.7 nM T61622 CPR8Q2 44339874 IC50 = 1.8 nM T61622 CM4QS7 44339906 IC50 = 2.5 nM T61622 C95IKD 44339907 IC50 = 2.8 nM T61622 CD1K2W 44339967 IC50 = 1.2 nM T61622 CI6GJ4 44339968 IC50 = 1.15 nM T61622 CKO06D 44340179 IC50 = 28.5 nM T61622 C1IC4W 44340209 IC50 = 2.4 nM T61622 C81HET 44340210 IC50 = 2.9 nM T61622 CQZ9M4 44340211 IC50 = 1.5 nM T61622 CH6T1N 44340274 IC50 = 140000 nM T61622 CF6BE8 44340280 IC50 > 330000 nM T61622 CK6UB4 44340295 IC50 > 330000 nM T61622 C5ED3O 44340316 IC50 = 320 nM T61622 CI58YE 44340320 IC50 > 330000 nM T61622 CMA36T 44340351 IC50 > 330000 nM T61622 CE4FL1 44340366 IC50 = 140000 nM T61622 CWJ8T7 44342184 IC50 = 4 nM T61622 CX65JI 44342269 IC50 = 500 nM T61622 C1VBW4 44342328 IC50 = 7.1 nM T61622 CGN5F1 44342372 Ki = 14 nM T61622 CP26NT 44342415 IC50 > 100 nM T61622 CP0VH2 44344886 IC50 = 175 nM T61622 C2US9C 44344887 IC50 = 130 nM T61622 CI54PU 44344919 IC50 = 310 nM T61622 C80AOD 44344920 IC50 = 150 nM T61622 C35DFT 44344921 IC50 = 190 nM T61622 CA69LX 44344922 IC50 = 140 nM T61622 CU45CD 44344981 IC50 = 58 nM T61622 C85JED 44345011 IC50 = 130 nM T61622 CKI70N 44345017 IC50 = 37 nM T61622 C4GH5E 44345110 IC50 = 770 nM T61622 C6CSJ5 44345111 IC50 = 140 nM T61622 C15ZBX 44345134 IC50 = 9.3 nM T61622 CCH1S0 44345173 IC50 = 750 nM T61622 CV4XF3 44345978 Ki = 600 nM T61622 CRP0O7 44346071 Ki = 300 nM T61622 CRH37B 44346092 Ki = 2200 nM T61622 CS4BG9 44346190 Ki = 42000 nM T61622 C8REA2 44346212 Ki = 100 nM T61622 C3N7IX 44348175 IC50 = 2 nM T61622 CB1XL9 44348176 IC50 = 6 nM T61622 C0OKF2 44348192 IC50 = 6 nM T61622 CTX45E 44348205 IC50 > 10000 nM T61622 CUR3D1 44348281 IC50 = 12 nM T61622 CKZE51 44348283 IC50 = 70 nM T61622 C9IU2Z 44348284 IC50 = 25 nM T61622 C3X8OW 44348322 IC50 = 5.5 nM T61622 CHN3X9 44348347 IC50 = 19 nM T61622 CF0KG8 44348359 IC50 = 16 nM T61622 C8YNB0 44348360 IC50 = 580 nM T61622 CZG59X 44348361 IC50 = 86 nM T61622 C5PKI4 44348362 IC50 = 7.6 nM T61622 CK7N5G 44348374 IC50 = 10 nM T61622 CHB7I0 44348384 IC50 = 230 nM T61622 C79COH 44348397 IC50 = 1.3 nM T61622 CIQF16 44348409 IC50 = 2 nM T61622 C5SMA7 44348410 IC50 = 18 nM T61622 C49PQC 44348443 IC50 = 22 nM T61622 CKW0G8 44348444 IC50 = 3.9 nM T61622 CI1LT2 44348447 IC50 = 7 nM T61622 C0FH5T 44348448 IC50 = 170 nM T61622 CZY53B 44348461 IC50 = 330 nM T61622 CDT56I 44348560 IC50 = 58 nM T61622 CJ64NX 44348561 IC50 = 20000 nM T61622 CM14EV 44348562 IC50 = 200 nM T61622 CXAN73 44348563 IC50 = 1800 nM T61622 C1EON0 44348685 IC50 = 3.4 nM T61622 CLP2T5 44348731 IC50 = 840 nM T61622 C5KYX3 44348742 IC50 = 1.3 nM T61622 C3IE2T 44348754 IC50 = 0.23 nM T61622 C5F9CH 44349517 IC50 = 840 nM T61622 CBT7L1 44349729 IC50 = 22 nM T61622 CD04WU 44349845 IC50 = 7.7 nM T61622 C5Y1BL 44349856 IC50 = 4200 nM T61622 C5O0YJ 44349857 IC50 = 25 nM T61622 C2ERV4 44349858 IC50 = 1.7 nM T61622 C50YOI 44349930 IC50 = 290 nM T61622 CK1U6M 44349967 IC50 = 62 nM T61622 COW43J 44360355 IC50 = 2400 nM T61622 CLS4F9 44360627 IC50 = 170 nM T61622 CNU91L 44360632 IC50 = 0.99 nM T61622 C4D8VG 44360634 IC50 = 120 nM T61622 CNS7F1 44360947 IC50 = 7.4 nM T61622 CH6D8U 44361024 IC50 = 110 nM T61622 CX35ES 44362231 IC50 > 10000 nM T61622 CIPY68 44362240 IC50 > 10000 nM T61622 C0Q5WH 44363833 IC50 = 46 nM T61622 C8YD0L 44363870 IC50 = 20 nM T61622 CU2ID0 44364010 IC50 = 360 nM T61622 CMY8I6 44364011 IC50 = 4.8 nM T61622 CEY62L 44364013 IC50 = 130 nM T61622 C1N8CK 44364025 IC50 = 25 nM T61622 CGQ71A 44364036 IC50 = 2.8 nM T61622 C4S7WC 44364072 IC50 = 115 nM T61622 C6B8ZX 44364143 IC50 = 55 nM T61622 C93BFN 44364156 IC50 = 10.5 nM T61622 C56ZYD 44366609 IC50 = 2500 nM T61622 C57HTC 44366741 IC50 = 40000 nM T61622 CN5OS1 44366804 IC50 = 35000 nM T61622 CY2HR1 44367156 IC50 = 15000 nM T61622 CJ2UD7 44368300 IC50 = 2.4 nM T61622 CT0HM5 44368301 IC50 = 4.4 nM T61622 C7ZIA3 44368512 IC50 = 12 nM T61622 CK07AQ 44370533 Ki = 1900 nM T61622 CFB98M 44370558 Ki = 24400 nM T61622 CA2C1S 44370759 Ki = 10900 nM T61622 CN21DY 44370803 Ki = 960000 nM T61622 CS3J1U 44370809 Ki = 440000 nM T61622 CD4Y0P 44370862 Ki = 520000 nM T61622 CX04DV 44370882 Ki = 2440000 nM T61622 CX9MH7 44370888 Ki = 1520000 nM T61622 CK8A7X 44370946 Ki = 1010000 nM T61622 C9H8FM 44371769 IC50 = 7 nM T61622 C73LHB 44371838 IC50 = 1 nM T61622 C0URL7 44373078 IC50 = 27000 nM T61622 C6KTY2 44373080 IC50 = 25000 nM T61622 CWBN35 44373189 IC50 = 250 nM T61622 CWBS43 44373703 IC50 = 1700 nM T61622 CUI18E 44373751 IC50 = 1800 nM T61622 CEI0A9 44373752 IC50 = 440000 nM T61622 CJ8A5B 44373765 IC50 = 2500000 nM T61622 CPF53M 44373777 IC50 = 50 nM T61622 C7CQ5B 44373871 IC50 = 550000 nM T61622 C39JDE 44373872 IC50 = 5800 nM T61622 CW5OR4 44373895 IC50 = 360 nM T61622 CCG60J 44373896 IC50 = 18000 nM T61622 CM17YF 44373944 IC50 = 100000 nM T61622 CO4GH7 44373947 IC50 = 140000 nM T61622 C0UA4N 44373954 IC50 = 1600 nM T61622 CDC8A4 44373955 IC50 = 3000 nM T61622 CDX53F 44373956 IC50 = 2300 nM T61622 CHJR82 44373976 IC50 = 330000 nM T61622 C8J2OZ 44373977 IC50 = 1000000 nM T61622 C5UL2Y 44374163 IC50 = 4100 nM T61622 C3E2QB 44374717 IC50 = 1300 nM T61622 C4CYT6 44374718 IC50 = 770 nM T61622 CM1HG2 44379569 Ki = 2 nM T61622 C3LA2W 44379720 Ki = 212 nM T61622 C54XME 44380144 IC50 = 141 nM T61622 CM40KP 44380145 IC50 = 36 nM T61622 C3GAE6 44380165 IC50 = 8 nM T61622 CQ04EU 44380170 IC50 = 23 nM T61622 C5UXG1 44380294 IC50 = 2100 nM T61622 CV57JL 44380316 IC50 = 80 nM T61622 CA7OB5 44380355 IC50 = 391 nM T61622 CEL0N4 44380356 IC50 = 157 nM T61622 C5PU4L 44380425 IC50 = 6500 nM T61622 C6QA3J 44380426 IC50 = 1400 nM T61622 CQJA62 44380427 IC50 = 630 nM T61622 C6KG5E 44380462 IC50 = 186 nM T61622 CJ83GH 44380489 IC50 = 4400 nM T61622 CA5CL3 44380670 IC50 > 100000 nM T61622 CA2JS0 44380671 IC50 = 18000 nM T61622 CMV21I 44380689 IC50 = 23000 nM T61622 C6CRO3 44380690 IC50 = 21000 nM T61622 C5S2WQ 44380691 IC50 = 3800 nM T61622 CZ05IQ 44380692 IC50 = 8400 nM T61622 CFG2W4 44380693 IC50 = 1200 nM T61622 C98WBU 44380718 IC50 = 5400 nM T61622 C32UFC 44380725 IC50 = 4000 nM T61622 C3X5HV 44380726 IC50 = 6700 nM T61622 C9B7NW 44380727 IC50 = 23000 nM T61622 CE69LB 44380728 IC50 = 320 nM T61622 CNID52 44380729 IC50 = 530 nM T61622 CA0YP9 44380779 IC50 = 5600 nM T61622 CD18ZJ 44380804 IC50 = 11000 nM T61622 CR6D9U 44380805 IC50 = 470 nM T61622 C7UQP5 44380811 IC50 = 200 nM T61622 C9LN6R 44380812 IC50 = 3800 nM T61622 C0IWP9 44380813 IC50 = 4200 nM T61622 CST56C 44380814 IC50 = 3700 nM T61622 C1UO4M 44380860 IC50 = 90 nM T61622 CTJ9F5 44380904 IC50 = 22 nM T61622 CQ1NX5 44380905 IC50 = 61 nM T61622 CF27UT 44380911 IC50 = 1500 nM T61622 CT3WX8 44380912 IC50 = 1300 nM T61622 C3R6UP 44380916 IC50 = 640 nM T61622 CK2YJ9 44380917 IC50 = 87 nM T61622 CRPE14 44380918 IC50 = 0.84 nM T61622 CX7O1U 44380919 IC50 = 2.1 nM T61622 CT63IM 44380920 IC50 = 210 nM T61622 C6GWI0 44380935 IC50 = 18 nM T61622 C3B0AF 44380936 IC50 = 7000 nM T61622 CXRK90 44380986 IC50 = 13000 nM T61622 CDL8R5 44381002 IC50 = 9200 nM T61622 C3UQ8P 44381003 IC50 = 1100 nM T61622 CXQ1Z2 44381006 IC50 = 29000 nM T61622 CB8LJ5 44381007 IC50 = 3800 nM T61622 C4Q8RK 44381008 IC50 = 11000 nM T61622 CAV68G 44381009 IC50 = 26000 nM T61622 C62BUK 44381114 IC50 = 2000 nM T61622 CEY42U 44381115 IC50 = 7400 nM T61622 C2LXY6 44381132 IC50 = 6500 nM T61622 CI2AZ4 44381133 IC50 = 18000 nM T61622 CVHB27 44381134 IC50 = 10000 nM T61622 CJCD89 44381135 IC50 = 15000 nM T61622 C0XHK5 44381148 IC50 = 780 nM T61622 CK4N5Y 44382655 IC50 = 47 nM T61622 C5MTR9 44382895 IC50 = 1.5 nM T61622 CK4N3U 44382899 IC50 > 20000 nM T61622 CMB9W5 44383534 IC50 = 200 nM T61622 C6BY1K 44384695 IC50 = 3200 nM T61622 C4Z5HD 44384696 IC50 = 3000 nM T61622 CE08KV 44384916 IC50 = 63000 nM T61622 C1OH0S 44387610 IC50 = 2.6 nM T61622 C92SNH 44401869 IC50 = 820 nM T61622 C9WTE1 44401946 IC50 = 120 nM T61622 CAGR39 44401947 IC50 = 33 nM T61622 C5DBC8 44401948 IC50 = 64 nM T61622 CA4FZ2 44401949 IC50 = 35 nM T61622 CAG0X5 44401993 IC50 = 860 nM T61622 CE01CH 44402259 IC50 = 66 nM T61622 C4W9SM 44402889 IC50 = 1600 nM T61622 CO74DV 44402890 IC50 = 1200 nM T61622 C0KIX3 44402891 IC50 = 900 nM T61622 C0T9SK 44402892 IC50 = 600 nM T61622 CEKT68 44402896 IC50 = 7000 nM T61622 CR3YM2 44402897 IC50 = 6800 nM T61622 CUOQ70 44402898 IC50 = 3900 nM T61622 CR16ST 44402899 IC50 = 450 nM T61622 CW7ZL8 44402900 IC50 = 340 nM T61622 C5D8IO 44402901 IC50 = 330 nM T61622 C9PM6G 44402902 IC50 = 300 nM T61622 CZA65J 44402903 IC50 = 270 nM T61622 C5SX0H 44402904 IC50 = 270 nM T61622 CHQ62Y 44402905 IC50 = 410 nM T61622 CQB97U 44402906 IC50 = 410 nM T61622 C1BE3P 44402907 IC50 = 370 nM T61622 C93MAK 44402908 IC50 = 230 nM T61622 CQ0E5I 44402909 IC50 = 230 nM T61622 C3FO8U 44402910 IC50 = 180 nM T61622 C75GZY 44402911 IC50 = 180 nM T61622 C61JKS 44402912 IC50 = 140 nM T61622 C7OTD3 44402913 IC50 = 270 nM T61622 C4T2MS 44402914 IC50 = 260 nM T61622 C25XEI 44402915 IC50 = 250 nM T61622 C73GBN 44402916 IC50 > 1000 nM T61622 COY12D 44402917 IC50 = 5590 nM T61622 CK8DO5 44402918 IC50 = 594 nM T61622 CGV9Q4 44402919 IC50 > 10000 nM T61622 C3KRL6 44402932 IC50 > 1000 nM T61622 CXC57A 44421346 IC50 > 50000 nM T61622 CA71VT 44421347 IC50 > 50000 nM T61622 CU4B2Y 44441701 IC50 = 144000 nM T61622 C6QMY7 44441703 IC50 = 169000 nM T61622 C2JE8M 44441743 IC50 = 275000 nM T61622 CMA9Q1 44458240 IC50 = 27 nM T61622 C9AP4S 44458241 IC50 = 29 nM T61622 CU26KN 44458392 IC50 = 49 nM T61622 CP91BO 44458434 IC50 = 60 nM T61622 CC1G3O 44458516 IC50 = 2580 nM T61622 C7Q3YL 44458517 IC50 = 700 nM T61622 CFY07H 44458529 IC50 = 26 nM T61622 CWHK49 44458530 IC50 = 248 nM T61622 CAY9R1 44458536 IC50 = 29 nM T61622 C4XI1N 44458537 IC50 = 100 nM T61622 C4Q8IC 44458555 IC50 = 2490 nM T61622 CUX53E 44458557 IC50 = 10 nM T61622 CW8CH7 44458558 IC50 = 44 nM T61622 C9K0TD 44458559 IC50 = 58 nM T61622 CS4R5E 44458609 IC50 = 85 nM T61622 CV37LM 44458620 IC50 = 6.2 nM T61622 C5V4NP 44458641 IC50 = 350 nM T61622 C5X6BW 44458642 IC50 = 108 nM T61622 CEIG80 44458643 IC50 = 36 nM T61622 CO2CL6 44458648 IC50 = 19 nM T61622 C5YBR2 44458668 IC50 = 44 nM T61622 C6TI5Y 44458673 IC50 = 8000 nM T61622 CA15NF 44458674 IC50 = 90 nM T61622 CAK45D 44458675 IC50 = 40 nM T61622 C1DWF5 44458676 IC50 = 48 nM T61622 CA17GV 44458677 IC50 = 700 nM T61622 CP89ZQ 44458679 IC50 = 20 nM T61622 C7BS4A 44458680 IC50 = 39 nM T61622 CT5K3M 44458685 IC50 = 120 nM T61622 C7T6JM 44458698 IC50 = 3.3 nM T61622 CQT05J 44458699 IC50 = 3.2 nM T61622 CSY3V2 44458711 IC50 = 3000 nM T61622 CQ21GN 44458712 IC50 = 89 nM T61622 CCQ75B 44458713 IC50 = 87 nM T61622 C5GSF6 44458716 IC50 = 390 nM T61622 CWN90A 44458721 IC50 = 0.5 nM T61622 CBMA53 44458722 IC50 = 14 nM T61622 C75LRQ 44458723 IC50 = 350 nM T61622 C4Q6TY 44458727 IC50 = 740 nM T61622 CQ9R2C 44458728 IC50 = 5.4 nM T61622 CSF1V5 44458729 IC50 = 2.3 nM T61622 CDW1Z4 44458734 IC50 = 8.7 nM T61622 CAM30U 44458735 IC50 = 9 nM T61622 C3QPB5 44458759 IC50 = 10560 nM T61622 CX02JB 44458760 IC50 = 47 nM T61622 C9LUQ7 44458761 IC50 = 395 nM T61622 C1Q6IC 44458762 IC50 = 3.3 nM T61622 COTU50 44458777 IC50 = 12 nM T61622 CO3J1M 44458783 IC50 = 13 nM T61622 CM3EV2 44459558 IC50 = 10 nM T61622 CINT92 44459559 IC50 = 41 nM T61622 CIY8C9 44459577 IC50 = 100000 nM T61622 C9V6BS 44459578 IC50 = 400 nM T61622 CF9WM1 44459588 IC50 = 40 nM T61622 C2DO0W 44459589 IC50 = 20 nM T61622 CEC19S 44459615 IC50 = 4 nM T61622 CS2D8H 44459623 IC50 = 3 nM T61622 C09SOV 44459627 IC50 = 37 nM T61622 CJ08BE 44459628 IC50 = 170 nM T61622 C5KG2H 44459629 IC50 = 55 nM T61622 CT25RA 44459638 IC50 = 4 nM T61622 CJ5Q0U 44459639 IC50 = 8 nM T61622 C6IW5Y 44459652 IC50 = 20 nM T61622 CJV5K7 44459672 IC50 = 68000 nM T61622 C67INO 44459673 IC50 = 430 nM T61622 C4KW6O 44459674 IC50 > 100000 nM T61622 CB2F4O 44459682 IC50 = 6 nM T61622 CNL1P9 44459683 IC50 = 14 nM T61622 C9YNK5 44459684 IC50 = 38 nM T61622 C12QOD 44459691 IC50 = 30 nM T61622 C2KBG0 44459698 IC50 = 95 nM T61622 C2YC4T 44459699 IC50 = 34 nM T61622 C4A5JW 44459700 IC50 = 12 nM T61622 CF61BV 44459725 IC50 = 16 nM T61622 C1O4DE 44459812 IC50 = 220 nM T61622 CC6J1A 44459814 IC50 = 900 nM T61622 C17BAJ 44460211 IC50 = 52000 nM T61622 C5OCY4 44460212 IC50 = 420000 nM T61622 CGNH45 44460354 IC50 = 4.7 nM T61622 C2U4WQ 44460709 IC50 = 14 nM T61622 C5DLV4 44460710 IC50 = 23 nM T61622 CF2HZ0 44460711 IC50 = 110 nM T61622 C5AF6Q 44460733 IC50 = 5 nM T61622 C6WG7X 44460734 IC50 = 4.1 nM T61622 CNB71X 44460735 IC50 = 6400 nM T61622 CM0CA4 44460782 IC50 = 2200 nM T61622 CGWM79 44460858 IC50 = 15 nM T61622 C5O0RJ 44460859 IC50 = 3200 nM T61622 CGT38B 44462719 IC50 = 1 nM T61622 CJ39UE 44473168 IC50 = 2 nM T61622 CDZP10 44479308 IC50 = 0.62 nM T61622 CXJN29 44479309 IC50 = 0.32 nM T61622 C4Y5GO 44479310 IC50 = 0.64 nM T61622 CJ25FS 44479563 IC50 = 0.6 nM T61622 C4CPX0 44479566 IC50 = 0.24 nM T61622 CI7EX6 44479809 IC50 = 8.4 nM T61622 C1FTA7 44481065 IC50 = 2.3 nM T61622 CVW53Z 44481067 IC50 = 42 nM T61622 C5COJ1 44481316 IC50 = 0.3 nM T61622 C8TIN9 44481318 IC50 = 8 nM T61622 CC2Q0J 44481321 IC50 = 0.6 nM T61622 C13ZGK 44481860 IC50 = 1.4 nM T61622 CR3TH8 44481861 IC50 = 17 nM T61622 CW1ZR7 44481862 IC50 = 3 nM T61622 C8O9PY 44482139 IC50 = 7.1 nM T61622 CB0O7Y 44482409 IC50 = 1.7 nM T61622 C7XV2J 44512857 IC50 = 13 nM T61622 C8XR6S 44517739 IC50 = 7 nM T61622 CDB7V6 44517740 IC50 = 2 nM T61622 CB46WL 44543660 IC50 = 1.3 nM T61622 CIXZ18 44554894 IC50 = 0.84 nM T61622 C7D8TR 44574907 IC50 = 0.55 nM T61622 C14HVE 44574908 IC50 = 0.55 nM T61622 CJND70 44574909 IC50 = 1.8 nM T61622 C8XH4S 44574910 IC50 = 2.9 nM T61622 CLI15D 44574911 IC50 = 120 nM T61622 CWL9S3 44602422 IC50 = 5 nM T61622 CKG61X 44610811 IC50 = 0.8 nM T61622 C2YE7A 45254510 IC50 > 1000 nM T61622 C43HDC 45256109 IC50 > 3000 nM T61622 C2YW4K 45259745 Ki = 95000 nM T61622 C2MRP6 45263606 IC50 = 26 nM T61622 CX2QO0 45263613 IC50 = 6 nM T61622 CU52TY 45263614 IC50 = 0.9 nM T61622 C0DWK9 45263616 IC50 = 20 nM T61622 CR5D8N 45263620 IC50 = 13 nM T61622 CW03RP 45267708 IC50 = 100 nM T61622 CZQ2V3 45267713 IC50 = 300 nM T61622 C9CL5K 45267720 IC50 = 670 nM T61622 CWJ16O 45268578 IC50 = 2 nM T61622 C51UQS 45268584 IC50 = 6 nM T61622 CH5GP6 45269509 IC50 = 15 nM T61622 CK3JC4 45270275 IC50 = 1 nM T61622 CW19XB 45270278 IC50 = 13 nM T61622 C6F4RI 45271083 IC50 = 2 nM T61622 C9MEW8 45271093 IC50 = 8 nM T61622 CPZ1E6 45271101 IC50 > 100000 nM T61622 C2OPF3 45271109 IC50 = 1000 nM T61622 CZ9I0S 45272903 IC50 = 1 nM T61622 CEHP97 45273762 IC50 = 8 nM T61622 C67QLM 45482028 IC50 > 2046000 nM T61622 C0MBR6 45482029 IC50 > 1991000 nM T61622 CGU92Y 45482030 IC50 > 2117000 nM T61622 CRDO76 45482033 IC50 > 1935000 nM T61622 CDW9Y5 45482036 IC50 > 1990000 nM T61622 CIS49D 45482037 IC50 > 1663000 nM T61622 CHMZ65 45488102 IC50 = 59500 nM T61622 CH7SG2 45488107 IC50 = 13800 nM T61622 CH0W9R 45488121 IC50 = 23200 nM T61622 CE74UZ 46191161 IC50 = 0.48 nM T61622 C72VYT 46224856 IC50 = 2.5 nM T61622 CV64LO 46224857 IC50 = 2.1 nM T61622 CG16QK 46224892 IC50 = 2.7 nM T61622 CSN59O 46224924 IC50 = 2.1 nM T61622 CFG52L 46224925 IC50 = 0.87 nM T61622 CV24OD 46224926 IC50 = 0.58 nM T61622 CLHP57 46224954 IC50 = 2.9 nM T61622 CVEO46 46224955 IC50 = 0.47 nM T61622 CK1DQ9 46224980 IC50 = 14 nM T61622 C0HDB2 46225011 IC50 = 0.18 nM T61622 C8KLO3 46225012 IC50 = 46 nM T61622 CDR02T 46225013 IC50 = 2260 nM T61622 C4SI2B 46225036 IC50 = 46 nM T61622 C4X9CP 46225037 IC50 = 31 nM T61622 CM23JK 46225038 IC50 = 177 nM T61622 CI3N7E 46225071 IC50 = 17 nM T61622 CB50WQ 46225072 IC50 = 57 nM T61622 CF2L1U 46225073 IC50 = 21 nM T61622 CKYA39 46225147 IC50 = 0.23 nM T61622 CC36NU 46861797 IC50 = 1.7 nM T61622 C1XZ9A 46880050 IC50 = 1.37 nM T61622 C4YZI8 46880051 IC50 = 0.92 nM T61622 C07LAP 46880052 IC50 = 0.4 nM T61622 C32SNI 46880053 IC50 = 0.68 nM T61622 CF98CZ 46880054 IC50 = 1.1 nM T61622 CV7MW4 46880055 IC50 = 6.4 nM T61622 C7YC0K 46880056 IC50 = 170 nM T61622 C42XED 46880057 IC50 = 64 nM T61622 C9EQ1J 46880058 IC50 = 210 nM T61622 CL8K6G 46880059 IC50 = 0.55 nM T61622 CGH8L6 46880060 IC50 = 53 nM T61622 C3GT7H 46880061 IC50 = 31 nM T61622 CMA1P8 46880062 IC50 = 0.49 nM T61622 CBW9M5 46880063 IC50 = 0.74 nM T61622 CZ38CX 46880064 IC50 = 2 nM T61622 CDM27Q 46880065 IC50 = 330 nM T61622 CXV01F 46883797 IC50 = 0.26 nM T61622 CN5C0Y 46883798 IC50 = 0.09 nM T61622 CHF8B0 46883799 IC50 = 0.21 nM T61622 C8NK4H 46883800 IC50 = 0.19 nM T61622 C9UMT6 46883801 IC50 = 2.9 nM T61622 CGK06T 46883802 IC50 = 1.5 nM T61622 CZ0AI1 46883803 IC50 = 31 nM T61622 C86ADS 46883844 IC50 = 0.27 nM T61622 C5ZRV0 46883845 IC50 = 0.11 nM T61622 C0BJD3 46883846 IC50 = 0.09 nM T61622 CR8N2G 46883847 IC50 = 2.2 nM T61622 CG2LJ5 46883848 IC50 = 1.8 nM T61622 CIP28U 46884482 IC50 = 650 nM T61622 C0Z4FK 46905393 IC50 = 1.1 nM T61622 C2J6MS 46912134 IC50 = 91 nM T61622 C5XAF7 46912235 IC50 = 0.05 nM T61622 CO7GU8 46931232 IC50 = 3.8 nM T61622 C3D7FL 46931619 IC50 = 0.5 nM T61622 CW3L9K 46931735 IC50 = 0.5 nM T61622 C3M4LT 46931848 IC50 = 0.08 nM T61622 C9EG4R 46931852 IC50 = 4.8 nM T61622 CB84WK 46931947 IC50 = 3.52 nM T61622 CJMS30 46931948 IC50 = 11 nM T61622 CD4L1A 46931949 IC50 = 73.8 nM T61622 C2M1KO 46932044 IC50 = 402 nM T61622 C3QLC4 46932045 IC50 = 1213 nM T61622 CC91MK 46932046 IC50 = 2500 nM T61622 CQ91FA 46932047 IC50 = 3.7 nM T61622 C70QIV 46932048 IC50 = 0.21 nM T61622 CYCF24 46932049 IC50 = 27 nM T61622 C3O4MA 46932136 IC50 = 0.47 nM T61622 CF9YV2 46932138 IC50 = 0.06 nM T61622 COL7J6 46932139 IC50 = 0.36 nM T61622 CSMK50 46932141 IC50 = 166 nM T61622 C29RXO 46932234 IC50 = 0.17 nM T61622 CC0F4D 46932235 IC50 = 2.82 nM T61622 C8QB4Z 46932237 IC50 = 1333 nM T61622 CG2J9V 46932512 IC50 = 0.73 nM T61622 C2VZ7Q 46932514 IC50 = 0.26 nM T61622 C4PW3A 46932704 IC50 = 0.37 nM T61622 C82QKP 46932796 IC50 = 1.4 nM T61622 CDI36J 46944860 IC50 = 0.04 nM T61622 C03KOR 46945859 IC50 = 0.09 nM T61622 C3E1TK 49867581 IC50 = 2 nM T61622 CZV62M 49867582 IC50 = 5000 nM T61622 C1R5UC 50905013 IC50 = 0.11 nM T61622 C5C7JP 50913994 IC50 = 2.8 nM T61622 CMXA29 50914146 IC50 = 1.3 nM T61622 CT9C1J 50914303 IC50 = 2.1 nM T61622 CJ1Q4N 50914305 IC50 = 2.1 nM T61622 CQ0O8I 50914306 IC50 = 3.3 nM T61622 CR3N4T 50914448 IC50 = 1.8 nM T61622 C41KNA 50914449 IC50 = 2.4 nM T61622 C9HPZ1 50914590 IC50 = 1.6 nM T61622 CDI09M 52934690 IC50 = 1.3 nM T61622 CUV9B4 52934924 IC50 = 0.14 nM T61622 CQJG83 52940639 IC50 = 0.11 nM T61622 CV4FS6 52940640 IC50 = 0.24 nM T61622 CO2N1D 52940643 IC50 = 0.1 nM T61622 CJ6M8H 52940810 IC50 = 5900 nM T61622 CH4BC7 52940901 IC50 = 752 nM T61622 CH7DU8 52940938 IC50 = 11 nM T61622 CBK69R 52941025 IC50 = 122 nM T61622 C2MN7B 52941035 IC50 = 20 nM T61622 C1K4ZE 52941036 IC50 = 0.18 nM T61622 C0O1UN 52941434 IC50 = 1.7 nM T61622 CA0L6U 52941636 IC50 = 0.08 nM T61622 CSD3O6 52941670 IC50 = 44 nM T61622 CQ7E3H 52941681 IC50 = 0.3 nM T61622 CBX64O 52941835 IC50 = 3.7 nM T61622 CHIK04 52941836 IC50 = 0.11 nM T61622 CYV50Z 52941837 IC50 = 0.62 nM T61622 C80UVC 52941838 IC50 = 0.09 nM T61622 CQ6P9U 52941842 IC50 = 0.14 nM T61622 C50RFT 52942013 IC50 = 1600 nM T61622 CFIJ38 52942087 IC50 = 707 nM T61622 C4FUO1 52942136 IC50 = 773 nM T61622 C3G1WY 52942172 IC50 = 84 nM T61622 C1OJ9Y 52942257 IC50 = 1.4 nM T61622 CQ4HV5 52942286 IC50 = 3800 nM T61622 CYM20B 52942582 IC50 = 2.1 nM T61622 CL56WB 52942783 IC50 = 30.8 nM T61622 CHN91J 52942848 IC50 = 5600 nM T61622 C1CJL4 52942895 IC50 = 0.13 nM T61622 CYPW08 52942941 Ki = 1140000 nM T61622 CE42QS 52943065 IC50 = 0.05 nM T61622 C96YUQ 52943066 IC50 = 0.2 nM T61622 CLN71C 52943274 IC50 = 4500 nM T61622 CB8K0N 52943342 IC50 = 16 nM T61622 CU4Z8T 52943410 IC50 = 12 nM T61622 CRAI23 52944034 IC50 = 130 nM T61622 C34CRE 52944053 IC50 = 1350 nM T61622 CA1B4V 52944247 IC50 = 0.11 nM T61622 CLB56M 52944248 IC50 = 0.57 nM T61622 CU3A9E 52944254 IC50 = 0.7 nM T61622 CTGX03 52944414 IC50 = 20 nM T61622 CQPD40 52944421 IC50 = 5300 nM T61622 CO65EG 52944458 IC50 = 7300 nM T61622 CH0PY6 52944486 IC50 = 9350 nM T61622 CLK45V 52944495 IC50 = 360 nM T61622 C4NSB8 52944566 IC50 = 64 nM T61622 CD9B6W 52944597 IC50 = 6 nM T61622 C3RV8A 52944640 IC50 = 29 nM T61622 CEU86L 52944649 IC50 = 0.29 nM T61622 CX4Q1R 52945024 IC50 = 416 nM T61622 C9OE1C 52945179 IC50 = 0.97 nM T61622 C0AS8I 52945257 IC50 = 11 nM T61622 C8S3QJ 52945476 IC50 = 0.04 nM T61622 CH8CU5 52945477 IC50 = 35.3 nM T61622 CKE3O4 52945479 IC50 = 0.9 nM T61622 COHA73 52945778 IC50 = 63 nM T61622 CJ4N8B 52945779 IC50 = 4 nM T61622 CQBR69 52945900 IC50 = 4 nM T61622 C36ISZ 52945945 IC50 = 447 nM T61622 CEO8R7 52946288 IC50 = 614 nM T61622 CQ4V8R 52946545 IC50 = 8600 nM T61622 C96TSE 52946688 IC50 = 0.13 nM T61622 CW53TK 52946691 IC50 = 0.08 nM T61622 CKA6S8 52946692 IC50 = 0.05 nM T61622 CPA83X 52946869 IC50 = 34 nM T61622 C8PL7V 52946933 IC50 = 4970 nM T61622 C0BT7S 52946943 IC50 = 175 nM T61622 CR53VN 52946944 IC50 = 763 nM T61622 C2X1BL 52946960 IC50 = 24 nM T61622 CH2Q6N 52946997 IC50 = 4 nM T61622 CYP6W4 52947015 IC50 = 6460 nM T61622 CA68NY 52947115 IC50 = 4 nM T61622 C6WOV2 52947913 IC50 = 0.05 nM T61622 CAR13H 52947916 IC50 = 0.17 nM T61622 CIB68Q 52947917 IC50 = 0.21 nM T61622 CAV7K8 52948057 IC50 = 12.9 nM T61622 CB3NQ0 52948140 IC50 = 5900 nM T61622 CY34UI 52948154 IC50 = 6100 nM T61622 CKT0J6 52948174 IC50 = 8100 nM T61622 CB90WK 52948313 IC50 = 680 nM T61622 CAZH65 52948317 IC50 = 0.62 nM T61622 C8NM6Q 52948980 IC50 = 9000 nM T61622 C3A5UP 52949001 IC50 = 31 nM T61622 C82YEM 52949120 IC50 = 24 nM T61622 C4M1AF 52949144 IC50 = 0.31 nM T61622 C9OWB4 52949145 IC50 = 0.27 nM T61622 C1T5RL 52949146 IC50 = 0.28 nM T61622 CP5Y7K 52949379 IC50 = 0.18 nM T61622 C2XIY3 52949466 IC50 = 16600 nM T61622 C4ML3H 52949494 IC50 = 10.6 nM T61622 CU37SY 52949546 IC50 = 71 nM T61622 CHQ29U 52949576 IC50 = 0.5 nM T61622 CC79IA 52949577 IC50 = 1 nM T61622 C7GX0L 52949581 IC50 = 11 nM T61622 C2IB6A 52949598 IC50 = 2 nM T61622 CBU7N9 52950051 IC50 = 1.02 nM T61622 CPO5A7 52950127 IC50 = 10900 nM T61622 CNAF49 52950192 IC50 = 0.68 nM T61622 CB6PX1 53232388 IC50 = 1.3 nM T61622 CHLQ29 53232610 IC50 = 1.9 nM T61622 C5WQ2E 53232611 IC50 = 1.7 nM T61622 C7IJ2F 53232612 IC50 = 0.9 nM T61622 CCX5G2 53232721 IC50 = 1.4 nM T61622 CE0R8K 53232722 IC50 = 1.6 nM T61622 CC3R7S 53232723 IC50 = 1.1 nM T61622 C0NW2T 53232833 IC50 = 1.3 nM T61622 C5TK3Z 53301844 IC50 = 37 nM T61622 CQ87XN 53307874 IC50 < 0.02 nM T61622 CW4S5E 53307875 IC50 = 0.04 nM T61622 C7V1YI 53307876 IC50 = 0.06 nM T61622 C6QY4D 53307877 IC50 = 0.03 nM T61622 C68TEC 53307957 IC50 = 0.04 nM T61622 C3DIM5 53316912 Ki = 450 nM T61622 CQA2R7 53318217 Ki = 3.3 nM T61622 CZ89RV 53319354 IC50 = 0.2 nM T61622 CI4O5J 53320863 Ki = 94 nM T61622 C5AZH3 53322198 Ki = 34 nM T61622 CWUZ14 53322199 Ki = 340 nM T61622 C9O2CI 53324843 Ki > 5000 nM T61622 C61FYW 53326116 Ki = 130 nM T61622 CXY4G5 53326117 Ki = 940 nM T61622 CQV61H 53346499 IC50 = 226 nM T61622 C3HQF5 53357854 IC50 = 0.2 nM T61622 C2ZUV8 53357855 IC50 = 1.12 nM T61622 CYZ0F6 53379391 IC50 = 1.1 nM T61622 CR5Y0Q 53387513 IC50 = 189 nM T61622 C35JSC 53387514 IC50 = 328 nM T61622 C2KRP8 53387671 IC50 = 3 nM T61622 C95IRG 53387672 IC50 = 159 nM T61622 C6NOA7 53497561 IC50 = 0.42 nM T61622 CMDO43 54580283 IC50 = 5 nM T61622 C8S1LG 54581286 IC50 = 0.028 nM T61622 C4ZG3O 54581303 IC50 = 3 nM T61622 CI12NU 54584263 IC50 = 37 nM T61622 CY80OU 54584273 IC50 = 0.01 nM T61622 CZ3TB4 54585225 IC50 = 0.4 nM T61622 C6VQT3 54587171 IC50 = 0.022 nM T61622 CO19MR 54587173 IC50 = 2.1 nM T61622 CAH7Y1 54681312 IC50 > 10000 nM T61622 C3P8YE 54681383 IC50 > 10000 nM T61622 C3JNM1 54753101 IC50 = 1.3 nM T61622 CH3C2O 56657671 IC50 = 350 nM T61622 CYZ9A3 56657672 IC50 = 120 nM T61622 CF9DT7 56657673 IC50 = 6.5 nM T61622 CPSV93 56657710 IC50 = 3.5 nM T61622 CB54JD 56657941 IC50 = 517 nM T61622 C98KJV 56658187 IC50 = 98 nM T61622 CAS35R 56658190 IC50 > 5000 nM T61622 CV4N2C 56658319 IC50 = 98 nM T61622 CP04UI 56658320 IC50 = 231 nM T61622 C5IMP0 56658321 IC50 = 88 nM T61622 C7IS6T 56658322 IC50 = 80 nM T61622 CCV75H 56659181 IC50 = 11 nM T61622 C1IHZ4 56659182 IC50 = 3.7 nM T61622 CKE72P 56659183 IC50 = 5.2 nM T61622 CX46ZL 56659184 IC50 = 1.6 nM T61622 CN2GB5 56659185 IC50 = 1.1 nM T61622 C5NS9V 56659278 IC50 = 3.8 nM T61622 CXBH95 56659572 IC50 = 150 nM T61622 C2ABY4 56659668 IC50 = 4.85 nM T61622 C94USX 56659669 IC50 = 1.08 nM T61622 C9LB2W 56659670 IC50 = 1.15 nM T61622 CJZS68 56660076 IC50 = 0.8 nM T61622 CXSM32 56661192 IC50 = 49 nM T61622 CYL93H 56661194 IC50 = 170000 nM T61622 CIW90M 56661235 IC50 = 220 nM T61622 CM7G6Z 56661287 IC50 > 10000 nM T61622 CC4EB9 56661372 IC50 = 14 nM T61622 C7R1SN 56661689 IC50 = 1000 nM T61622 C2R9ZF 56661690 IC50 = 246 nM T61622 CW8JU7 56661691 IC50 = 455 nM T61622 CAEW49 56661692 IC50 = 110 nM T61622 CU8B3L 56661821 IC50 = 5060 nM T61622 C35BJX 56661822 IC50 = 396 nM T61622 C5WME2 56661823 IC50 = 170 nM T61622 C9ZOM2 56661824 IC50 = 6410 nM T61622 CB56XY 56661825 IC50 = 4670 nM T61622 CPHZ63 56661826 IC50 = 847 nM T61622 C2WPN0 56662683 IC50 = 420 nM T61622 CO6Z4P 56662684 IC50 = 195 nM T61622 CQM06L 56662685 IC50 = 1437 nM T61622 CRAT94 56662686 IC50 = 19 nM T61622 CF2R0K 56662687 IC50 = 2.1 nM T61622 CME1K7 56663526 IC50 = 61 nM T61622 CMI4D9 56663528 IC50 = 0.88 nM T61622 CWSX53 56664640 IC50 = 6200 nM T61622 CAZ78S 56664679 IC50 = 0.34 nM T61622 CQL20F 56664680 IC50 = 1.9 nM T61622 CRQY23 56664752 IC50 > 10000 nM T61622 CT7Y3B 56664903 IC50 = 850 nM T61622 C2NO4Z 56665114 IC50 = 107 nM T61622 CZSK39 56665115 IC50 = 15 nM T61622 CJDV92 56665116 IC50 = 1460 nM T61622 C6WX2I 56665117 IC50 = 60 nM T61622 C4G3EH 56665118 IC50 = 143 nM T61622 C54JQI 56665119 IC50 = 1180 nM T61622 C9YSP2 56665120 IC50 = 285 nM T61622 CEU36P 56665121 IC50 = 80 nM T61622 CV3B1Q 56665122 IC50 = 9 nM T61622 CP42VF 56665262 IC50 = 15 nM T61622 COS79D 56665263 IC50 = 181 nM T61622 CP1VC2 56665264 IC50 = 150 nM T61622 CZ1B7A 56665265 IC50 = 73 nM T61622 CQK85J 56665266 IC50 = 99 nM T61622 CUGC46 56666142 IC50 = 7.1 nM T61622 CPJM20 56666143 IC50 = 1.9 nM T61622 CUF46J 56666144 IC50 = 1.8 nM T61622 C76VCW 56666710 IC50 = 0.91 nM T61622 CGQ23I 56666711 IC50 = 0.36 nM T61622 CLF45N 56666970 IC50 = 9 nM T61622 CYVP10 56668100 IC50 = 8.5 nM T61622 C9TOE4 56668164 IC50 > 10000 nM T61622 CGC89H 56668554 IC50 = 320 nM T61622 CU18DE 56668555 IC50 = 3260 nM T61622 CBA79U 56668556 IC50 = 1100 nM T61622 CY4OD3 56668561 IC50 = 322 nM T61622 CIX2U8 56668562 IC50 = 290 nM T61622 C10PMU 56668563 IC50 = 57 nM T61622 CHZJ93 56668564 IC50 = 3 nM T61622 C5L9DF 56668718 IC50 = 504 nM T61622 C9Z6CA 56668719 IC50 = 116 nM T61622 CVGX27 56668837 IC50 = 12 nM T61622 C87NUY 56669541 IC50 = 1.2 nM T61622 CVU7S3 56669542 IC50 = 4700 nM T61622 C7D1CY 56669543 IC50 = 2.5 nM T61622 C9YMP8 56669622 IC50 = 1.6 nM T61622 CF06GH 56669910 IC50 = 460 nM T61622 CLB4M9 56670001 IC50 = 2.17 nM T61622 CC7FH3 56670429 IC50 = 0.06 nM T61622 CH2V0E 56671530 IC50 = 26 nM T61622 CM0JT7 56671533 IC50 = 6000 nM T61622 CRF9M6 56671625 IC50 > 10000 nM T61622 C8HRV9 56671819 IC50 = 423 nM T61622 C37TWO 56672053 IC50 = 11 nM T61622 CRDC15 56672055 IC50 = 310 nM T61622 CML2G4 56672056 IC50 = 70 nM T61622 CHC0Z7 56672057 IC50 = 14 nM T61622 CRQ85K 56672193 IC50 = 1830 nM T61622 CUN75I 56672194 IC50 = 89 nM T61622 CQGT36 56672195 IC50 = 218 nM T61622 CGWR57 56672805 IC50 = 0.26 nM T61622 CY95OX 56673062 IC50 = 8.8 nM T61622 CWUI93 56673063 IC50 = 2900 nM T61622 C39ADI 56673420 IC50 = 4.9 nM T61622 C19GOU 56673914 IC50 = 0.4 nM T61622 C7KJ9C 56675009 IC50 = 0.7 nM T61622 CZ05JR 56675057 IC50 > 10000 nM T61622 CL2JS3 56675215 IC50 = 112 nM T61622 CBP35O 56675442 IC50 = 55 nM T61622 CY09IV 56675443 IC50 = 61 nM T61622 C2HT4X 56675444 IC50 = 152 nM T61622 C6UEW1 56675445 IC50 = 6630 nM T61622 C3TNI7 56675580 IC50 = 86 nM T61622 CA51PD 56675581 IC50 = 650 nM T61622 CJ46TM 56676148 IC50 = 0.33 nM T61622 CY5E1U 56676373 IC50 = 2.7 nM T61622 CORN57 56676374 IC50 = 2.1 nM T61622 COI26V 56676375 IC50 = 1.4 nM T61622 C1UJ2C 56676376 IC50 = 1.6 nM T61622 CW86SU 56676730 IC50 = 45 nM T61622 COV8P5 56676820 IC50 = 4.13 nM T61622 C3GVN5 56676821 IC50 = 0.83 nM T61622 CV79CF 56677248 IC50 = 0.07 nM T61622 C2DY5F 56678284 IC50 = 0.82 nM T61622 CN2O0D 56678324 IC50 = 17 nM T61622 C94ASY 56678325 IC50 = 1.2 nM T61622 C82SRZ 56678327 IC50 = 58 nM T61622 C0QUG6 56678526 IC50 = 320 nM T61622 CV4A6X 56678527 IC50 = 5 nM T61622 C63NMC 56678778 IC50 = 692 nM T61622 COWE13 56678779 IC50 = 513 nM T61622 CUM8Q3 56678780 IC50 = 202 nM T61622 CHEW40 56678781 IC50 = 4 nM T61622 CRC5Y1 56678782 IC50 = 390 nM T61622 CTF35V 56678783 IC50 = 2710 nM T61622 C9MBV2 56678906 IC50 = 1850 nM T61622 CI5J2O 56678907 IC50 = 24 nM T61622 C3HEB8 56679079 IC50 = 1.1 nM T61622 CQ7KJ4 56679708 IC50 = 596 nM T61622 CTS97E 56679709 IC50 > 5000 nM T61622 CXU86O 56679710 IC50 = 23 nM T61622 C1E2AG 56679711 IC50 = 10 nM T61622 CE3F9I 56680150 IC50 = 0.81 nM T61622 CIB7O5 56680151 IC50 = 1.02 nM T61622 CCW34H 56680290 IC50 = 1.64 nM T61622 C8UK2V 56680291 IC50 = 2.88 nM T61622 CPW21N 56681634 IC50 = 2500 nM T61622 C3WU2Y 56681670 IC50 = 2 nM T61622 C8SW4E 56682095 IC50 = 37 nM T61622 CFY13W 56682096 IC50 = 154 nM T61622 CV9X8C 56682097 IC50 = 4090 nM T61622 CKT0B1 56682098 IC50 = 80 nM T61622 C1NJ9U 56682099 IC50 = 694 nM T61622 CGP23S 56682222 IC50 = 1230 nM T61622 C7UQO9 56682223 IC50 = 186 nM T61622 C9FE8V 56682777 Ki = 0.043 nM T61622 CLHN14 56683031 IC50 = 126 nM T61622 CCA89K 56683032 IC50 = 20 nM T61622 CHF79L 56683033 IC50 = 0.7 nM T61622 CUM62D 56683034 IC50 = 2.3 nM T61622 CP9G8Z 56683392 IC50 = 25 nM T61622 CG6A2R 56683486 IC50 = 1.48 nM T61622 C2QKL9 56683615 IC50 = 3.84 nM T61622 CGR7Y1 56683616 IC50 = 4.23 nM T61622 C01ORB 56683617 IC50 = 0.79 nM T61622 CH92EZ 56683889 IC50 = 81 nM T61622 CY1W2Q 56683890 IC50 = 0.05 nM T61622 C7SIV2 56834949 IC50 = 106000 nM T61622 CK7HJ8 56837192 IC50 = 0.07 nM T61622 CP8H0D 56962365 IC50 = 2.1 nM T61622 C1TR4E 56963091 IC50 = 0.27 nM T61622 CM37LJ 57390221 IC50 = 0.26 nM T61622 C58KFP 57390222 IC50 = 1.5 nM T61622 CSCB73 57390223 IC50 = 0.38 nM T61622 CP8D5L 57390807 IC50 = 90 nM T61622 CDJC72 57390808 IC50 = 5 nM T61622 CE03ZS 57390809 IC50 = 0.7 nM T61622 C41VBK 57392010 IC50 = 135 nM T61622 CT96ZS 57392011 IC50 = 42 nM T61622 CB6C4T 57392012 IC50 = 0.11 nM T61622 CCZJ34 57392013 IC50 = 0.07 nM T61622 CP48ZB 57392014 IC50 = 0.36 nM T61622 C16PSG 57392623 IC50 = 150 nM T61622 CFM8E5 57392624 IC50 = 0.08 nM T61622 CH97QF 57393726 IC50 = 0.17 nM T61622 CM80PV 57393727 IC50 = 0.05 nM T61622 CJE1N0 57393728 IC50 = 130 nM T61622 CWC2E8 57393729 IC50 = 3.4 nM T61622 C1GT2K 57394201 IC50 = 537.03 nM T61622 CHA2Q7 57394339 IC50 = 7.1 nM T61622 CS8M9I 57394340 IC50 = 3.7 nM T61622 CLP4Z8 57394341 IC50 = 0.5 nM T61622 C8PWV4 57394342 IC50 = 0.18 nM T61622 C16OJD 57394343 IC50 = 0.8 nM T61622 C0AJM8 57394344 IC50 = 4.2 nM T61622 C6HR3Q 57394345 IC50 = 0.5 nM T61622 C6VQ7I 57395454 IC50 = 14 nM T61622 CFE6D4 57395455 IC50 = 0.09 nM T61622 CHX4Z7 57396095 IC50 = 1900 nM T61622 CRS39Y 57396096 IC50 = 0.3 nM T61622 CLEH95 57396097 IC50 = 1.5 nM T61622 C4NVE2 57396098 IC50 = 0.6 nM T61622 C7PT9Q 57396099 IC50 = 0.3 nM T61622 C23WQH 57396100 IC50 = 0.05 nM T61622 C9WB0G 57397294 IC50 = 0.24 nM T61622 C7GJ6H 57397295 IC50 = 0.1 nM T61622 C7ML8N 57397296 IC50 = 0.04 nM T61622 CLR02T 57397297 IC50 = 0.45 nM T61622 CEYO28 57397298 IC50 = 14 nM T61622 CB20QV 57397299 IC50 = 0.76 nM T61622 CH4Z3O 57397916 IC50 = 40 nM T61622 CI4PT1 57398835 IC50 = 229.09 nM T61622 CH25BK 57398981 IC50 = 2.7 nM T61622 C4EY3H 57398982 IC50 = 2.2 nM T61622 CNY94K 57398983 IC50 = 1.5 nM T61622 CG1D3L 57398984 IC50 = 0.08 nM T61622 C2J7GK 57398992 IC50 = 2.5 nM T61622 CB42RN 57399556 IC50 = 5.2 nM T61622 C9IXS8 57400698 IC50 = 0.15 nM T61622 C3XQ0F 57401188 IC50 = 426.58 nM T61622 CUYK04 57401306 IC50 = 390 nM T61622 CSQK78 57401307 IC50 = 1.3 nM T61622 C8GC4D 57401308 IC50 < 0.01 nM T61622 CFL71K 57401309 IC50 = 49 nM T61622 CJQ89O 57401397 IC50 = 1 nM T61622 C2PXA4 57402998 IC50 = 15.85 nM T61622 CQ1ZV2 57403067 IC50 = 0.2 nM T61622 CBU2H4 57404035 IC50 = 6.457 nM T61622 CX7M2I 57519702 IC50 = 1.4 nM T61622 CN0CF4 57544848 IC50 = 0.27 nM T61622 C9FH4B 57790981 IC50 = 0.3 nM T61622 CNG70S 58017410 IC50 = 2.7 nM T61622 C5B0RJ 58083331 IC50 = 4.3 nM T61622 C1C6OS 58083336 IC50 = 0.26 nM T61622 C6DZ0X 58083358 IC50 = 0.14 nM T61622 CQ7XG8 58355122 IC50 = 3.3 nM T61622 CJON31 58355176 IC50 = 0.59 nM T61622 CJZD63 58355221 IC50 = 1.1 nM T61622 C2ST9V 58355241 IC50 = 0.66 nM T61622 CP8T7G 58355269 IC50 = 0.4 nM T61622 CSK0N7 58355353 IC50 > 10 nM T61622 CIM0A7 58355366 IC50 = 0.81 nM T61622 C5QA3E 58355435 IC50 = 2.6 nM T61622 CV0O6P 58355440 IC50 = 0.9 nM T61622 CAQZ34 58355464 IC50 = 3.3 nM T61622 C7JX8A 58355480 IC50 = 0.63 nM T61622 CXD42B 58355489 IC50 = 1.2 nM T61622 CAW15G 58355526 IC50 = 0.32 nM T61622 C2YF1B 58355540 IC50 = 1.2 nM T61622 CX69UP 58355573 IC50 = 1.1 nM T61622 C7BQ1H 58355668 IC50 = 16 nM T61622 C1YZ3E 58355693 IC50 = 0.16 nM T61622 CI26UZ 59201574 IC50 = 0.33 nM T61622 CJ5D0B 59271966 IC50 = 30 nM T61622 C1M2FH 59271973 IC50 = 65 nM T61622 C2BGW6 59271984 IC50 = 8 nM T61622 CY5IM3 59271988 IC50 = 300 nM T61622 CO3SQ2 59271989 IC50 = 150 nM T61622 C65KTJ 59271991 IC50 = 150 nM T61622 C2PJ4N 59271992 IC50 = 30 nM T61622 CUE79I 59272004 IC50 = 8 nM T61622 CK0V2L 59272005 IC50 = 20 nM T61622 CXG7L0 59272011 IC50 = 60 nM T61622 C1V5EC 59272020 IC50 = 60 nM T61622 CZCV65 59272024 IC50 = 90 nM T61622 CC8L6W 59272028 IC50 = 170 nM T61622 C1XI3N 59272033 IC50 = 100 nM T61622 C7AOL2 59272040 IC50 = 20 nM T61622 CI86EV 59272041 IC50 = 25 nM T61622 CN7EQ9 59272046 IC50 = 300 nM T61622 C8YHJ2 59272059 IC50 = 1000 nM T61622 CTK95R 59272061 IC50 = 1150 nM T61622 C25NCB 59272065 IC50 = 15 nM T61622 C9EY7K 59272074 IC50 = 10 nM T61622 C8G6SZ 59272087 IC50 = 550 nM T61622 C8KZ3J 59272093 IC50 = 15 nM T61622 C9ZN2U 59272130 IC50 = 90 nM T61622 CF4C5R 59272140 IC50 = 350 nM T61622 C10MUY 59272165 IC50 = 200 nM T61622 CP68JF 59272188 IC50 = 65 nM T61622 C49VES 59272189 IC50 = 90 nM T61622 CK8GF7 59272204 IC50 = 2250 nM T61622 C8Z0MJ 59272210 IC50 = 450 nM T61622 C4QO0N 59272218 IC50 = 200 nM T61622 CTQ42U 59272220 IC50 = 85 nM T61622 C63MCF 59272222 IC50 = 2050 nM T61622 CBR20V 59272225 IC50 = 450 nM T61622 C1MTZ2 59272228 IC50 = 35 nM T61622 CBJ7W1 59272237 IC50 = 9200 nM T61622 CJ9PT3 59272251 IC50 = 70 nM T61622 C0S6UA 59272254 IC50 = 145 nM T61622 CCD08Z 59272264 IC50 = 250 nM T61622 C2QBE7 59272265 IC50 = 500 nM T61622 CQV86Z 59272290 IC50 = 50 nM T61622 CKO4S7 59272298 IC50 = 65 nM T61622 C7AWY5 59563537 IC50 = 1.6 nM T61622 C9PL4C 59620419 IC50 = 1.3 nM T61622 C1W6VL 59620422 IC50 = 1 nM T61622 CHY1P5 59620426 IC50 = 3.2 nM T61622 CK13WB 59620428 IC50 = 320 nM T61622 CY15CD 59620457 IC50 = 2.5 nM T61622 CT52DP 59620461 IC50 = 2 nM T61622 CNW27P 59620483 IC50 = 16 nM T61622 C0V2QS 59625209 IC50 = 1.4 nM T61622 C68XQI 59625236 IC50 = 11000 nM T61622 C30PKZ 59625306 IC50 = 0.039 nM T61622 C7QV2E 59625307 IC50 = 5.2 nM T61622 CF1C0N 59625336 IC50 = 3.3 nM T61622 CF9OR8 59625393 IC50 = 38000 nM T61622 CQME32 59625516 IC50 = 1.2 nM T61622 C8SID6 59625541 IC50 = 5.4 nM T61622 CY3O0B 59625584 IC50 = 4.6 nM T61622 CQW7A8 60149247 Ki = 0.6 nM T61622 CUBM51 60162599 IC50 = 1.4 nM T61622 C0Y6NM 60162601 IC50 = 1.7 nM T61622 CM48NK 60162861 IC50 = 1.3 nM T61622 CD3VT4 66645361 IC50 = 1.4 nM T61622 CM67TK 66645388 IC50 = 2.1 nM T61622 CA13UN 66645431 IC50 = 4.2 nM T61622 C2H5XA 66645466 IC50 = 2.4 nM T61622 CO80EM 66645472 IC50 = 3.1 nM T61622 CV3X0Y 66645480 IC50 = 2.4 nM T61622 CGD28B 66645492 IC50 = 1.4 nM T61622 C8XD9Y 66645544 IC50 = 1.7 nM T61622 CHQ6C3 66645605 IC50 = 2 nM T61622 CMD1O0 66645608 IC50 = 2.2 nM T61622 CNG30I 66645615 IC50 = 1.4 nM T61622 C7EUF0 66645650 IC50 = 2.9 nM T61622 CK7R5J 66645652 IC50 = 2.1 nM T61622 CZ7I8R 66645660 IC50 = 2 nM T61622 CJ9G3V 66645690 IC50 = 1.2 nM T61622 CI1QA0 66645695 IC50 = 1.4 nM T61622 CX0R5H 66645736 IC50 = 3 nM T61622 C8L3RW 66645739 IC50 = 5.5 nM T61622 CE2A0J 66645756 IC50 = 1.7 nM T61622 CJK4X8 66645801 IC50 = 2.4 nM T61622 CD21UF 66645804 IC50 = 1 nM T61622 C9NA2C 66645815 IC50 = 1.7 nM T61622 CD24FC 66645833 IC50 = 1.9 nM T61622 C89YJQ 66645837 IC50 = 1.6 nM T61622 C47LDH 66645839 IC50 = 2 nM T61622 C5R3LZ 66645840 IC50 = 2.1 nM T61622 CPM25W 66645852 IC50 = 1.4 nM T61622 CPIO91 66645862 IC50 = 1.8 nM T61622 CGXL53 66645879 IC50 = 1.9 nM T61622 C96ZTE 66645882 IC50 = 1 nM T61622 C90ZQM 66645894 IC50 = 1.6 nM T61622 CK2I0X 66645985 IC50 = 1.8 nM T61622 CLGK95 66647367 IC50 = 2.1 nM T61622 CPW29C 68411962 IC50 = 3.1 nM T61622 C61SJG 68412618 IC50 = 0.6 nM T61622 C30WPU 68417067 IC50 = 0.3 nM T61622 CWA06X 68431518 IC50 = 1.2 nM T61622 CL10ZC 68432247 IC50 = 2.1 nM T61622 CA1S5U 68432286 IC50 = 0.58 nM T61622 CJC3S1 68432392 IC50 = 3.4 nM T61622 C2LXQ0 68433634 IC50 = 4.5 nM T61622 CMEA13 68445580 IC50 = 4100 nM T61622 CYSU75 68446051 IC50 = 1700 nM T61622 CX2KA4 68446370 IC50 = 1900 nM T61622 CAB4M3 68447092 IC50 = 250 nM T61622 C0VRQ1 68447156 IC50 = 7700 nM T61622 CEFY74 68448300 IC50 = 9800 nM T61622 C56CFA 68448803 IC50 = 25 nM T61622 CNI8V4 68785998 IC50 = 5 nM T61622 CX4VN5 69918384 IC50 = 1 nM T61622 C2HJ6K 69918387 IC50 = 2.1 nM T61622 CDQE76 70132509 Ki = 82 nM T61622 CO36JZ 70679349 IC50 = 406 nM T61622 C3Z5WO 70679350 IC50 = 7.7 nM T61622 CJ5UQ0 70679351 IC50 = 1.6 nM T61622 CB5W9M 70682025 IC50 = 370 nM T61622 CCQ2O1 70685489 IC50 = 2.2 nM T61622 CWQ6I5 70685707 IC50 = 0.31 nM T61622 CB01GM 70685709 IC50 = 2.5 nM T61622 CFT32Y 70685711 IC50 = 30 nM T61622 CD3J1G 70686280 IC50 = 400 nM T61622 C7RL0K 70686282 IC50 = 170 nM T61622 C9V6ML 70687502 IC50 = 0.22 nM T61622 CF07JR 70688397 IC50 = 130 nM T61622 CTEB57 70689883 IC50 = 1.8 nM T61622 C1O9EY 70689886 IC50 = 46 nM T61622 CN7ZK4 70689896 IC50 = 2.2 nM T61622 C7DWK0 70692597 IC50 = 1.4 nM T61622 C8HF6X 70694089 IC50 = 1.9 nM T61622 CDX5Y8 70694090 IC50 = 27 nM T61622 CD71IT 70694091 IC50 = 0.7 nM T61622 C89HIX 70694640 IC50 = 3.3 nM T61622 CTUQ03 70696214 Ki = 0.16 nM T61622 C1OEY9 71449049 IC50 = 95 nM T61622 C09CPY 71450425 IC50 = 69000 nM T61622 C6AFS0 71450829 IC50 = 8 nM T61622 CUM28A 71450965 IC50 = 43 nM T61622 CK0QB5 71450997 IC50 = 120 nM T61622 C1Y2CP 71452222 IC50 = 2.3 nM T61622 CE63GJ 71452681 IC50 > 10000 nM T61622 CMBW70 71452682 IC50 = 1400 nM T61622 CZ7K8X 71454446 IC50 < 10 nM T61622 CY3E5Z 71454448 IC50 > 1000 nM T61622 C62TRZ 71454451 IC50 > 10000 nM T61622 CUC93B 71455789 IC50 = 2700 nM T61622 CZ21OI 71455790 IC50 > 100000 nM T61622 CXIF96 71456221 IC50 = 20 nM T61622 CUO92T 71457568 IC50 = 0.29 nM T61622 CF9BU4 71458001 IC50 = 500 nM T61622 CXTK53 71458023 IC50 = 1 nM T61622 C5W9VD 71459919 IC50 = 2700 nM T61622 CD4X9I 71461234 IC50 = 8.4 nM T61622 C1V3AF 71461589 IC50 = 100 nM T61622 CK2N9F 71461611 IC50 > 10000 nM T61622 C0F5VB 71461612 IC50 > 10000 nM T61622 CH8O2Y 71461613 IC50 = 660 nM T61622 C2U1YX 71461692 IC50 = 2700 nM T61622 C3HP6U 71461725 IC50 = 3.9 nM T61622 C6HX9K 71462969 IC50 > 1000 nM T61622 CIEM86 71462971 IC50 = 2.5 nM T61622 CG9WQ0 71601779 IC50 = 500 nM T61622 CWM6L8 71659968 IC50 = 97 nM T61622 CS4Q1N 71659995 IC50 = 16 nM T61622 C7A3RJ 71660026 IC50 = 2.4 nM T61622 CMR5W1 71660065 IC50 = 3.2 nM T61622 C5GAX2 71660067 IC50 = 1.4 nM T61622 C9ANB0 71660107 IC50 = 1.9 nM T61622 CE57CA 71660109 IC50 = 2 nM T61622 CI5Z9W 71660111 IC50 = 0.9 nM T61622 CJ01PL 71660147 IC50 = 1 nM T61622 C5KM3O 71660149 IC50 = 1.7 nM T61622 C3C1HX 71660151 IC50 = 6.7 nM T61622 C0FD5G 71660153 IC50 = 5.6 nM T61622 C9IOF7 71660189 IC50 = 3.8 nM T61622 CA5G8X 71660191 IC50 = 1 nM T61622 CA2CT1 71660193 IC50 = 1.1 nM T61622 C1V3PC 71660195 IC50 = 1.1 nM T61622 CCN54Y 71660315 IC50 = 1.6 nM T61622 C4G9RK 71716082 IC50 = 10000 nM T61622 CS0TR2 71716182 IC50 > 100 nM T61622 C4Y2FP 71716697 IC50 = 14 nM T61622 CGL09W 71717896 IC50 = 64.57 nM T61622 CUV52W 71717999 IC50 > 30000 nM T61622 C4WF6J 71718000 IC50 > 100 nM T61622 CBL04J 71718014 IC50 = 450 nM T61622 C5RIE0 71719857 IC50 = 14000 nM T61622 C9CLH7 71738394 Ki = 2.2 nM T61622 CYO91H 71738790 Ki = 2 nM T61622 CY65HG 71738908 Ki = 86 nM T61622 CN2V1S 71738909 Ki = 56 nM T61622 CAF2Y0 71738915 Ki = 44 nM T61622 CFW3T4 72164471 IC50 = 2.3 nM T61622 C62RTH 72164473 IC50 = 5.2 nM T61622 CM7K5U 72164590 IC50 = 1.1 nM T61622 C7XN4A 72164592 IC50 = 1.9 nM T61622 CT0Y2X 73345600 IC50 > 1000000 nM T61622 CXZ79P 73345601 IC50 = 27 nM T61622 CXST85 73345602 IC50 = 8 nM T61622 C8VL7I 73345714 Ki = 230000 nM T61622 C1K4FG 73345715 Ki = 230000 nM T61622 CF9GN5 73346989 IC50 > 100000 nM T61622 CI9U1N 73347122 IC50 = 100000 nM T61622 CYI20L 73347123 IC50 = 240 nM T61622 C87EVS 73347124 IC50 = 67 nM T61622 CK57ED 73347125 IC50 = 30 nM T61622 CY4C6V 73347126 IC50 = 3900 nM T61622 C7P2KI 73350150 Ki = 300000 nM T61622 CG6OJ8 73350489 IC50 = 2 nM T61622 CGQ5A1 73351540 IC50 = 430 nM T61622 C9R0WY 73351707 IC50 = 30 nM T61622 CJQ6O7 73351708 IC50 = 900 nM T61622 CD56UH 73351709 IC50 = 10 nM T61622 C5W8NY 73354699 IC50 = 49 nM T61622 C7I3ZW 73355790 IC50 = 26 nM T61622 C3N9SR 76871907 IC50 > 30000 nM T61622 CTVA19 76871908 IC50 > 30000 nM T61622 CLP57R 78350457 IC50 = 200 nM T61622 C8VMX7 88643446 IC50 = 750 nM T61622 CHL64A 89818372 Ki = 19 nM T61622 CZD0B6 89818377 Ki = 15 nM T61622 C54DVB 89818383 Ki = 6 nM T61622 CVCR46 90285136 IC50 = 16000 nM T61622 CD79MA 90285610 IC50 > 30000 nM T61622 CA7P0E 90285921 IC50 = 8400 nM T61622 C2ANE7 90285955 IC50 = 27000 nM T61622 C79LYP 90294431 IC50 = 8700 nM T61622 C7VUB6 90662791 IC50 = 0.52 nM T61622 C6K1ZI 90662792 IC50 = 1.7 nM T61622 CG1KP2 90662793 IC50 = 34 nM T61622 COE97J 90662794 IC50 = 12 nM T61622 CLQ0R8 90662797 IC50 = 24 nM T61622 CC8KW4 90662798 IC50 = 68 nM T61622 C7DFX1 90662799 IC50 = 190 nM T61622 C8EW0S 90662800 IC50 = 0.57 nM T61622 C2XYG5 90662801 IC50 = 730 nM T61622 CU5J9L 90662802 IC50 = 6800 nM T61622 C0O1YD 90662803 IC50 = 340 nM T61622 CM4FR2 90662804 IC50 = 720 nM T61622 C48GAQ 90662805 IC50 = 13 nM T61622 CJ0U6M 90662806 IC50 = 2.5 nM T61622 CX21HP 90662807 IC50 = 450 nM T61622 C5STY4 90662809 IC50 = 0.65 nM T61622 C3PCB6 90662810 IC50 = 100 nM T61622 CY57EX 90662811 IC50 > 10000 nM T61622 C3VFY9 90662815 IC50 = 1.3 nM T61622 C4MC3Z 90662828 IC50 = 5.5 nM T61622 CM3LN7 90662829 IC50 = 20 nM T61622 C8PGE4 90662830 IC50 = 6 nM T61622 C4F2SH 90662831 IC50 = 300 nM T61622 CCD60A 90662832 IC50 = 10 nM T61622 CAXM53 90662833 IC50 = 100 nM T61622 C81WSM 90662836 IC50 = 8 nM T61622 CT30HZ 90662853 IC50 = 1 nM T61622 CT6XY4 90662860 IC50 = 2.5 nM T61622 CQ2PW0 90662884 IC50 = 120.23 nM T61622 C3PL6O 90662886 IC50 = 257.04 nM T61622 CL5Q7J 90662887 IC50 = 173.78 nM T61622 CP6WG7 90662888 IC50 = 1412.54 nM T61622 CO7A9K 90662889 IC50 = 251.19 nM T61622 C9VJB7 90662890 IC50 = 151.36 nM T61622 CH41NW 90662891 IC50 = 112.2 nM T61622 CK6O3U 90662892 IC50 = 41.69 nM T61622 CI93VN 90662893 IC50 = 1412.54 nM T61622 CBC36R 90662894 IC50 = 1202.26 nM T61622 CKYP08 90662896 IC50 = 316.23 nM T61622 C8X2GB 90662899 IC50 = 10000 nM T61622 CUHS97 90662900 IC50 = 436.52 nM T61622 C2R6WF 90662901 IC50 = 316.23 nM T61622 C2L1XI 90662902 IC50 = 489.78 nM T61622 C2RVD0 90662903 IC50 = 37.15 nM T61622 CX96PZ 90662904 IC50 = 93.33 nM T61622 CLTQ23 90663143 IC50 = 440 nM T61622 C5HX7B 90663144 IC50 = 190 nM T61622 CZM05A 90663145 IC50 = 316.23 nM T61622 C4XG7S 90663147 IC50 = 480 nM T61622 CK6FW7 90663148 IC50 = 140 nM T61622 C8WGS1 90663150 IC50 = 15000 nM T61622 CQ3FH5 90663151 IC50 = 110 nM T61622 C1ZC6A 90663153 IC50 > 10000 nM T61622 C8OPU2 90663154 IC50 = 180 nM T61622 C1VN9T 90663157 IC50 > 10000 nM T61622 C7O3YT 90663158 IC50 = 30.2 nM T61622 CK3GT4 90663159 IC50 = 770 nM T61622 CEWO48 90663160 IC50 = 470 nM T61622 CNV03J 90663162 IC50 = 260 nM T61622 C98IHU 90663163 IC50 = 51.29 nM T61622 CB3PN9 90663171 IC50 = 250 nM T61622 C8ZUS3 90663172 IC50 = 350 nM T61622 CFN4D6 90663173 IC50 = 1000 nM T61622 CJ3OE1 90663174 IC50 = 750 nM T61622 CY2O8H 90663175 IC50 = 30 nM T61622 C4TWG7 90663237 IC50 = 0.6 nM T61622 CK0T2Y 90663376 IC50 = 50 nM T61622 CY3BW8 90663426 IC50 = 80 nM T61622 C50LJW 90663427 IC50 = 350 nM T61622 C0X9VU 90663428 IC50 = 20 nM T61622 CQOW40 90663430 IC50 = 39 nM T61622 C4NC7D 90663431 IC50 = 4000 nM T61622 CDYK59 90663432 IC50 = 90 nM T61622 CR0F1S 90663433 IC50 = 5100 nM T61622 C5UF1E 90663434 IC50 = 50 nM T61622 CYV6C8 90663435 IC50 = 47 nM T61622 CDX95P 90663436 IC50 = 1500 nM T61622 C5AH7F 90663437 IC50 = 72 nM T61622 C6KBR1 90663438 IC50 = 1500 nM T61622 C54DKP 90663439 IC50 = 400 nM T61622 C20KYN 90663440 IC50 = 2 nM T61622 C8EL7G 90663441 IC50 = 36 nM T61622 CVX0K3 90663442 IC50 = 43 nM T61622 CQ9L8M 90663443 IC50 = 3.5 nM T61622 CU95MY 90663450 IC50 = 1500 nM T61622 C8L5NV 90663452 IC50 = 50 nM T61622 C4U1JS 90663454 IC50 = 900 nM T61622 CH5P9L 90663455 IC50 = 120 nM T61622 CM6D8R 90663456 IC50 = 6 nM T61622 CQX08P 90663458 IC50 = 4 nM T61622 C7JD3U 90663459 IC50 = 20 nM T61622 C42KGZ 90663460 IC50 = 15 nM T61622 CBC6Y2 90663461 IC50 = 15 nM T61622 C1X9CA 90663462 IC50 = 15 nM T61622 CAHC43 90663463 IC50 = 30 nM T61622 CFUV68 90663464 IC50 = 35 nM T61622 C19IHV 90663465 IC50 = 600 nM T61622 CI09AK 90663466 IC50 = 10 nM T61622 CH9QP2 90663467 IC50 = 100 nM T61622 CSTC60 90663478 IC50 = 0.41 nM T61622 CT0C2A 90663480 IC50 = 0.66 nM T61622 C37MPE 90663482 IC50 = 0.28 nM T61622 CWE6B2 90663483 IC50 = 1.2 nM T61622 C7BX4L 90663485 IC50 = 0.45 nM T61622 CZ0X6P 90663498 Ki = 980000 nM T61622 CMAV52 90663499 Ki = 530000 nM T61622 CI14RZ 90663501 Ki = 670000 nM T61622 CP26UM 90663558 IC50 = 1000 nM T61622 CR3IC7 90663561 IC50 = 220 nM T61622 CN0B5T 90663562 IC50 = 3100 nM T61622 CCK5Q8 90663667 IC50 > 10000 nM T61622 CH82QG 90663676 IC50 = 34 nM T61622 C5C1EG 90663744 IC50 = 350 nM T61622 CKQ59S 90663745 IC50 = 1500 nM T61622 CJ1HU2 90663747 IC50 = 200 nM T61622 C52WKI 90663748 IC50 = 1000 nM T61622 C0Y2VG 90663749 IC50 = 4500 nM T61622 CLP9N2 90663750 IC50 = 10000 nM T61622 C0Y9PS 90663752 IC50 = 8000 nM T61622 C3N9UQ 90663753 IC50 = 960 nM T61622 CH9NJ1 90663754 IC50 = 81 nM T61622 CTW95C 90663757 IC50 = 7000 nM T61622 C74CDI 90663759 IC50 = 7000 nM T61622 C31JHO 90663762 IC50 = 600 nM T61622 CR7PM1 90663763 IC50 = 150 nM T61622 CAI58J 90663764 IC50 = 600 nM T61622 CW9DP0 90663768 IC50 = 3500 nM T61622 C9A5EX 90663769 IC50 = 1000 nM T61622 CTI3B6 90663771 IC50 = 800 nM T61622 C3LSW5 90663772 IC50 = 3000 nM T61622 CM73RZ 90663774 IC50 = 1500 nM T61622 C8LE7T 90663775 IC50 = 2000 nM T61622 CDI34J 90663776 IC50 = 1500 nM T61622 C4IJB6 90663777 IC50 = 500 nM T61622 C9X5RE 90663778 IC50 = 40 nM T61622 CJDO91 90663779 IC50 = 13 nM T61622 CMU5G2 90663780 IC50 = 90 nM T61622 CWZ5J1 90663782 IC50 = 1500 nM T61622 CBQ83Y 90663783 IC50 = 650 nM T61622 C5Q1GZ 90663828 IC50 = 1.7 nM T61622 CGW8V6 90663903 IC50 = 10000 nM T61622 C08QUP 90663904 IC50 = 100 nM T61622 CXCZ23 90663923 IC50 = 1.6 nM T61622 C1AWR4 90663924 IC50 = 40 nM T61622 CYQT26 90663934 Ki = 0.026 nM T61622 CKF9Z5 90663935 Ki = 3.6 nM T61622 CW5N0T 90663936 Ki = 14 nM T61622 CO60DJ 90663937 Ki = 580 nM T61622 CS6AI3 90663938 IC50 = 3.2 nM T61622 CW5XN9 90663939 Ki = 4100 nM T61622 CZC30I 90663940 Ki = 49 nM T61622 CR9LP8 90663941 IC50 = 100 nM T61622 CA72BY 90663942 Ki = 1.1 nM T61622 CL9D4Z 90663943 Ki = 0.88 nM T61622 C24JSQ 90663944 Ki = 0.52 nM T61622 CJB1D9 90663972 IC50 = 6000 nM T61622 CCK1H6 90664754 Ki = 900000 nM T61622 CJK38A 90664755 Ki = 740000 nM T61622 C9ATU5 90664759 Ki = 80000 nM T61622 CL5SW6 90713674 IC50 = 360 nM T61622 CT9B0E 91349601 IC50 = 6.3 nM T61622 C9ZY5P 91664005 IC50 = 80 nM T61622 C72FWD 91929322 IC50 = 1.1 nM T61622 CM4TS0 118576345 IC50 = 13000 nM T61622 CRNF04 118709230 IC50 = 1.1 nM T61622 C1M5PS 118709231 IC50 = 4 nM T61622 CV9QT4 118709233 IC50 = 1200 nM T61622 C86WUH 118709234 IC50 = 2600 nM T61622 C54NSW 118709235 IC50 = 300 nM T61622 C2RIB0 118709236 IC50 = 2 nM T61622 CARX10 118709238 IC50 = 0.3 nM T61622 CQ65IH 118709240 IC50 = 0.4 nM T61622 CG96QP 118709241 IC50 = 6 nM T61622 C8QO1J 118709242 IC50 = 0.2 nM T61622 CBK73W 118709243 IC50 = 0.6 nM T61622 C35GDB 118709244 IC50 = 2 nM T61622 CI9Q7O 118709245 IC50 = 0.6 nM T61622 CD0B1Z 118709246 IC50 = 0.2 nM T61622 CQ5NK9 118709822 IC50 > 30000 nM T61622 C4VDW0 118709823 IC50 > 30000 nM T61622 CDK81L 118709824 IC50 > 30000 nM T61622 CQM10N 118709825 IC50 > 30000 nM T61622 CXQD06 118709826 IC50 > 30000 nM T61622 CMZO04 118709827 IC50 > 30000 nM T61622 C86DZI 118709828 IC50 > 30000 nM T61622 C5MES8 118709829 IC50 = 20000 nM T61622 CAWM98 118709830 IC50 > 30000 nM T61622 C8ZHV3 118718102 IC50 = 55 nM T61622 C37ATR 118718104 IC50 = 0.3 nM T61622 C1M8DO 118718334 IC50 > 10000 nM T61622 CH5GL0 118718335 IC50 > 10000 nM T61622 C5LYJ6 118718337 IC50 = 470 nM T61622 C01DCW 118718338 IC50 > 10000 nM T61622 CALQ08 118718339 IC50 = 200 nM T61622 CVR3K7 118718350 IC50 = 3.5 nM T61622 CCO8B9 118718351 IC50 = 5.5 nM T61622 CI6W9F 118718352 Ki = 16 nM T61622 CW2K1B 118718353 Ki = 99 nM T61622 C1SVN3 118718354 Ki = 9 nM T61622 CIJ23K 118718355 Ki = 1100 nM T61622 C0EQ3L 118718356 Ki = 1700 nM T61622 CPOA29 118718365 Ki = 8 nM T61622 C4L8YU 118718714 IC50 = 85 nM T61622 C31RXA 118718818 IC50 = 20 nM T61622 C65AYZ 118718849 IC50 = 1.4 nM T61622 CSV4X5 118718870 Ki = 600000 nM T61622 CI85SC 118718871 Ki = 1780000 nM T61622 CYZ1B2 118727797 IC50 = 1670 nM T61622 C61QUC 118727798 IC50 = 730 nM T61622 CF68NZ 118727799 IC50 = 570 nM T61622 C4QNE1 118727800 IC50 = 850 nM T61622 CJW98I 118727801 IC50 = 1200 nM T61622 C7P9IU 118727802 IC50 = 5850 nM T61622 CN0G9R 118727803 IC50 = 300 nM T61622 CM7F6N 118727804 IC50 = 145 nM T61622 C5V3LE 118727805 IC50 = 200 nM T61622 CTE27B 118727806 IC50 = 2650 nM T61622 CUG74R 118727807 IC50 = 350 nM T61622 C97EMT 118727808 IC50 = 500 nM T61622 CD9U8R 118728410 Ki = 420 nM T61622 C5EQL1 118728570 IC50 = 180 nM T61622 CHR03X 118728571 IC50 = 55 nM T61622 CHW6Z4 118730134 IC50 = 3150 nM T61622 CZ78VI 118730135 IC50 = 350 nM T61622 CN1L7X 118730136 IC50 = 35 nM T61622 CFE7I9 118730137 IC50 = 20 nM T61622 C0HCB7 118730138 IC50 = 30 nM T61622 CJ2LQ7 118730139 IC50 = 9 nM T61622 C2GYF8 118730140 IC50 = 80 nM T61622 CELZ36 118866105 IC50 = 678000 nM T61622 C9M2WU 118866986 IC50 = 214000 nM T61622 CA9I7V 122194986 IC50 = 2.2 nM T61622 CV74AL 122194987 IC50 = 1.5 nM T61622 C1GF5H 122194988 IC50 = 34 nM T61622 C4C9MA 122194989 IC50 = 9.2 nM T61622 C6QTE5 122194991 IC50 = 9.8 nM T61622 C8EU2F 122194993 IC50 = 16.1 nM T61622 C1EKX4 122194995 IC50 = 12.4 nM T61622 CFN2I0 122194997 IC50 = 9.8 nM T61622 CYWL41 122194999 IC50 = 12.3 nM T61622 C4P7NB 122195001 IC50 = 10.2 nM T61622 CNU9Z8 122195003 IC50 = 13.4 nM T61622 CW1L7S 122195005 IC50 = 11.2 nM T61622 C2H5LV 122195007 IC50 = 15.5 nM T61622 CP62HJ 122195009 IC50 = 1.8 nM T61622 CP9I5L 122195011 IC50 = 8.5 nM T61622 C3GZA1 122195013 IC50 = 12.1 nM T61622 CV8QD0 122195015 IC50 = 11.5 nM T61622 C9M2VF 122195016 IC50 = 27.7 nM T61622 CHO7Y5 122195018 IC50 = 7.2 nM T61622 CPQH52 122195020 IC50 = 4.4 nM T61622 CTL1E2 122195022 IC50 = 11 nM T61622 CEZ56B 122195024 IC50 = 2.6 nM T61622 CWD89F 122195026 IC50 = 30 nM T61622 CH8OA4 122195028 IC50 = 15.2 nM T61622 CJL29G 122195030 IC50 = 33.7 nM T61622 C2O4LC 122195032 IC50 = 20.9 nM T61622 CCX7J5 122195034 IC50 = 1.6 nM T61622 CD4TJ3 122195036 IC50 = 7 nM T61622 C0EBH2 122195038 IC50 = 5.8 nM T61622 CRW1V4 122195040 IC50 = 17.1 nM T61622 C9AQN0 122195042 IC50 = 5 nM T61622 C8KM4W 122195044 IC50 = 13.1 nM T61622 CYKC32 122195046 IC50 = 1.5 nM T61622 CA6M5D 122195048 IC50 = 0.9 nM T61622 CLZ95N 122195050 IC50 = 0.7 nM T61622 C9Q2CL 122195052 IC50 = 1.1 nM T61622 CYQ23O 122195054 IC50 = 5.2 nM T61622 CHZB31 122195175 IC50 = 1.9 nM T61622 CBN51T 122195177 IC50 = 2.1 nM T61622 C5SQD7 122195179 IC50 = 2.7 nM T61622 CT6I3D 122195181 IC50 = 1 nM T61622 C4E2BU 122195183 IC50 = 1.1 nM T61622 CZD27X 132576081 IC50 = 491 nM T61622 C81IZS 132576082 IC50 = 500 nM T61622 CJL8W0 132576085 IC50 = 267 nM T61622 C63GWQ 132576086 IC50 = 69 nM T61622 CO2C3G 132585207 IC50 = 60 nM T61622 C4SJ1H 134141867 IC50 > 100000 nM T61622 C5HW0E 134144122 IC50 > 100000 nM T61622 CMRG25 134148766 IC50 = 140 nM T61622 CDRQ58 134152301 IC50 = 11000 nM T61622 C41DMR 134153166 IC50 = 73 nM T61622 CI1D7K 135875806 IC50 > 100000 nM T61622 CT1PK0 137632707 IC50 = 3370 nM T61622 CT1HB0 137638006 IC50 = 220 nM T61622 CY87JR 137638441 IC50 = 10200 nM T61622 COS4A9 137638535 IC50 = 1330 nM T61622 CRCO70 137640700 IC50 = 8260 nM T61622 C9Y4CM 137643002 IC50 = 360 nM T61622 C78UMY 137643003 IC50 = 121 nM T61622 CF75VD 137644746 IC50 = 1930 nM T61622 CSO9X3 137645468 IC50 = 45 nM T61622 CGX4B6 137646982 IC50 = 110 nM T61622 C7CSV6 137648833 IC50 = 7760 nM T61622 COYG97 137649952 IC50 = 8530 nM T61622 CD6FZ8 137650764 IC50 > 100000 nM T61622 C0QH2C 137653879 IC50 = 16800 nM T61622 C1MU5S 137653940 IC50 = 230 nM T61622 CB8Z9A 137654036 IC50 = 29200 nM T61622 C7DUA6 137654249 IC50 = 124000 nM T61622 CM45UH 137659567 IC50 = 3900 nM T61622 CNZU76 137660084 IC50 = 4520 nM T61622 C07TZL 145960467 IC50 > 100 nM T61622 CLIB76 145960838 IC50 = 35 nM T61622 C94OEX 145963289 IC50 = 2 nM T61622 C1CI2E 145963621 IC50 > 100 nM T61622 C7KD1V 145963758 IC50 = 630 nM T61622 CP56WZ 145963814 IC50 = 63 nM T61622 CEHK80 145963888 IC50 = 1.6 nM T61622 CLCO35 145963926 IC50 = 2 nM T61622 CYR72D 145963953 IC50 = 6.3 nM T61622 CNL1Y3 145963959 IC50 = 1000 nM T61622 CQA98S 145964789 IC50 = 16 nM T61622 CH6LC3 145964950 IC50 = 25 nM T61622 C6DZ1B 145965322 IC50 = 100 nM T61622 C1X3GZ 145966339 IC50 = 25 nM T61622 CC5S7D 145966340 IC50 = 320 nM T61622 C27KCT 145967479 IC50 = 1.3 nM T61622 CW5NY1 145967571 IC50 = 630 nM T61622 C9WH1E 145971784 IC50 = 2000 nM T61622 C25HJM 145971817 IC50 = 126 nM T61622 C4SM1J 145972774 IC50 = 3.2 nM T61622 CZ6A8N 145973086 IC50 = 2 nM T61622 CP02SN 145974180 IC50 = 6.3 nM T61622 C6Q7NJ 145974481 IC50 = 80 nM T61622 C0Q2NJ 145974673 IC50 = 2 nM T61622 CBL0F9 145975681 IC50 = 800 nM T61622 CF9W6A 145976587 IC50 = 40 nM T61622 C0IQV7 145977447 IC50 = 0.6 nM T61622 CYUB59 145978346 IC50 = 20 nM T61622 CY56OH 52945480 IC50 = 0.12 nM T61622 D01FJQ 44346213 Ki = 1000 nM T61622 D04QIA 9851682 IC50 = 0.039 nM T61622 D08BRJ 44346214 Ki = 4000 nM T61622 D09PZT 44297826 Ki = 1.5 nM T61622 D09SOY 15054176 IC50 = 9600 nM T61622 D0E5QB 52945901 IC50 = 0.06 nM T61622 D0K0OY 44346192 Ki = 800 nM T61622 D0KK6A 15126552 IC50 = 0.3 nM T61622 D0P6RT 10078814 IC50 = 1.2 nM T61622 D0P7NP 52948369 IC50 = 39 nM T61622 D0Y5IQ 44255320 IC50 = 50000 nM T56923 D00QKI 9865554 IC50 < 1 nM T56923 D00XBC 46861584 IC50 > 10000 nM T56923 D02JXG 9841667 IC50 = 10 nM T56923 D0LJ1B 9838712 IC50 = 1 nM T56923 D0O2XQ 11256587 IC50 > 10000 nM T56923 D0SN7I 10479502 IC50 = 5.1 nM T56923 D0F6WV 3854666 IC50 = 22 nM T56923 D03PDY 9887803 IC50 = 1.995 nM T56923 CO25SK 314241 IC50 > 30000 nM T56923 CF2H1L 990571 IC50 = 7800 nM T56923 CJV6X0 1105988 IC50 = 7600 nM T56923 CQAM15 1316559 IC50 = 6300 nM T56923 CY6S5I 1485055 IC50 = 2000 nM T56923 C0J1MS 4130676 IC50 > 30000 nM T56923 C9A8HM 4614441 IC50 > 30000 nM T56923 C7FT9O 9795327 IC50 = 1000 nM T56923 CUL5O7 9796076 IC50 = 3500 nM T56923 C6JH4S 9817855 IC50 = 1000 nM T56923 CR9VN5 9821417 IC50 = 15 nM T56923 C95KOI 9841701 IC50 = 14 nM T56923 C1KC6I 9842742 IC50 = 7 nM T56923 CK0H7P 9849040 IC50 = 110 nM T56923 C6ZXL9 9862533 IC50 = 3500 nM T56923 CAN73G 9868309 IC50 = 12 nM T56923 CJ0Q4K 9879541 IC50 = 3 nM T56923 CBI7Q4 9880342 IC50 = 22 nM T56923 C64ICF 9881570 IC50 = 4200 nM T56923 C7QGC3 9882303 IC50 = 890 nM T56923 CR9E5I 9883149 IC50 = 130 nM T56923 CR7ZN9 9884184 IC50 = 670 nM T56923 C29QKT 9885174 IC50 = 51 nM T56923 CDRB69 9885291 IC50 = 120 nM T56923 CCI9Y7 9888410 IC50 = 7 nM T56923 C0ND7U 9903068 IC50 = 220 nM T56923 CMWH46 9903859 IC50 = 1400 nM T56923 C6WPC0 9904302 IC50 = 1400 nM T56923 C41GVY 9910064 IC50 = 12.59 nM T56923 C5C7OU 9912703 IC50 = 5 nM T56923 C1REX8 9927727 IC50 < 28 nM T56923 CR6QI5 9928389 IC50 = 26 nM T56923 CRS37U 9946476 IC50 = 100 nM T56923 CJ89FT 9949617 IC50 = 350 nM T56923 CGV32C 9950107 IC50 = 350 nM T56923 CEC1R6 9951571 IC50 = 63 nM T56923 CYZT87 9953415 IC50 = 6 nM T56923 C91RTG 9956238 IC50 > 10000 nM T56923 CJV62S 9956678 IC50 = 0.7943 nM T56923 C4OKE6 9966255 IC50 = 32 nM T56923 CIDB47 9966717 IC50 = 10 nM T56923 CN56WL 9967031 IC50 = 130 nM T56923 CNAI53 9968028 IC50 = 15 nM T56923 C49SOU 9969306 IC50 = 125.89 nM T56923 CTDS90 9969483 IC50 = 90 nM T56923 C4MJ6R 9978981 Ki = 2 nM T56923 CRIG15 10003645 IC50 = 3.981 nM T56923 C1L2WF 10018018 IC50 = 1200 nM T56923 CE58ON 10027494 Ki = 4 nM T56923 CT97AZ 10050534 IC50 = 7.943 nM T56923 CLX3C1 10072431 IC50 = 5.012 nM T56923 CL7B2W 10072910 IC50 = 7.943 nM T56923 CUT41K 10112905 Ki = 20 nM T56923 CR0ZQ6 10127252 Ki = 10 nM T56923 CI3HK1 10134701 IC50 = 2 nM T56923 C3EVF9 10136860 Ki = 9 nM T56923 CNPV45 10143778 IC50 = 18 nM T56923 CP31MV 10150526 IC50 = 3.8 nM T56923 CG86FS 10150721 Ki = 4 nM T56923 CNU3L1 10154731 IC50 = 850 nM T56923 CNE95T 10155713 Ki = 25 nM T56923 C8RIM2 10161021 Ki = 20 nM T56923 CX9G0K 10179343 IC50 = 37 nM T56923 CRD2Z1 10180509 Ki = 11 nM T56923 CL5PT7 10186524 IC50 = 20 nM T56923 CTU8G7 10194831 Ki = 14 nM T56923 CU62YN 10200147 IC50 = 280 nM T56923 CG2F7V 10200589 Ki = 4 nM T56923 CR6X8O 10201676 IC50 = 4.9 nM T56923 CQR49K 10221030 IC50 = 7700 nM T56923 CIE61W 10222206 IC50 = 32 nM T56923 C59YEV 10224934 Ki = 18 nM T56923 CO0DS9 10224935 Ki = 10 nM T56923 CK14RC 10225736 Ki = 12 nM T56923 CV14ZH 10230576 Ki = 20 nM T56923 CD50IY 10237849 Ki = 1 nM T56923 CY8U6H 10237959 Ki = 3 nM T56923 C0C1GZ 10238257 Ki = 5 nM T56923 CXV73N 10252538 Ki = 3 nM T56923 C4L2TP 10252630 Ki = 4 nM T56923 CXO2N6 10263767 IC50 = 25000 nM T56923 C7M8NX 10267982 IC50 = 42 nM T56923 C3D9UQ 10268731 IC50 = 400 nM T56923 CKF0U3 10268984 IC50 = 8 nM T56923 CSZ71D 10269706 IC50 = 10 nM T56923 C3JON0 10270791 IC50 > 20000 nM T56923 CK49NQ 10272003 IC50 > 10000 nM T56923 C96NCK 10272255 Ki = 5 nM T56923 COJ5R3 10293087 Ki = 28 nM T56923 C1U2KT 10293321 IC50 = 5 nM T56923 CR17PX 10294353 IC50 = 6.2 nM T56923 CG9ZT6 10299249 Ki = 27 nM T56923 CLXR40 10309077 IC50 = 171 nM T56923 CKHY86 10310100 Ki = 1 nM T56923 CTWQ06 10343142 Ki = 4 nM T56923 CK2YO5 10345330 IC50 = 12.59 nM T56923 CL4G6W 10389383 IC50 = 30 nM T56923 CF9T6H 10411524 Ki = 3 nM T56923 C2CAD9 10412163 Ki = 6 nM T56923 C8LIQ4 10478354 Ki = 2 nM T56923 CKNU49 10479451 IC50 = 2.512 nM T56923 C3R7XL 10481927 Ki = 9 nM T56923 CI2SN0 11222420 IC50 = 81 nM T56923 CA39QR 11227406 IC50 > 10000 nM T56923 C20CDG 11245544 IC50 = 22 nM T56923 CQ6KW0 11272103 IC50 = 10000 nM T56923 CJS9C0 11304851 IC50 = 54 nM T56923 C1A5ET 11329244 IC50 = 10000 nM T56923 C7FS9V 11336278 IC50 = 5200 nM T56923 CL24DX 11371755 IC50 = 520 nM T56923 C70AVD 11440492 IC50 = 3.981 nM T56923 C0TEF4 11599650 IC50 = 0.631 nM T56923 C6H5VS 11625425 IC50 = 14 nM T56923 CD25ZL 11635447 Ki = 25 nM T56923 C96SCW 11656697 Ki = 44 nM T56923 CA1NU5 11750288 IC50 = 26 nM T56923 CC81AE 11754699 IC50 = 3.981 nM T56923 C8FEG4 11857486 Ki = 1360 nM T56923 CH3SY4 11857488 Ki = 210 nM T56923 C34JBI 11857680 IC50 = 13 nM T56923 CY8H4R 11858153 Ki = 21 nM T56923 C4PTK6 11858154 IC50 = 1 nM T56923 C7I5WK 11964579 Ki > 100000 nM T56923 C12JFO 11964663 Ki = 2100 nM T56923 CA98QX 11964664 Ki = 1400 nM T56923 C6JVN1 11965767 Ki = 2800 nM T56923 CM0W9F 12073809 IC50 = 4.5 nM T56923 C7D3MZ 12073810 IC50 = 1 nM T56923 CR74KQ 12229851 IC50 = 2400 nM T56923 CM74ZD 16098478 IC50 = 244 nM T56923 CAYQ40 16098479 IC50 = 234 nM T56923 C5X7MU 16098480 IC50 = 5 nM T56923 CQGO53 16098481 IC50 = 5.4 nM T56923 CR4AX9 16098482 IC50 = 6.2 nM T56923 CLC6F4 16098484 IC50 = 236 nM T56923 CFX6N0 16098485 IC50 = 17 nM T56923 C1BXN5 16098486 Ki = 5 nM T56923 CH2S4D 16098487 IC50 = 3.6 nM T56923 CUPD35 16098488 IC50 = 3.8 nM T56923 CEF6N1 16126703 IC50 = 29 nM T56923 CQ9G4U 17903294 IC50 = 2000 nM T56923 C9W0GF 17903299 IC50 = 450 nM T56923 CN1S5J 17903304 IC50 = 800 nM T56923 CUB38J 17903305 IC50 = 2000 nM T56923 CU8Y1N 17903311 IC50 = 450 nM T56923 CWLS87 17903316 IC50 = 2300 nM T56923 CYS69U 17903317 IC50 = 410 nM T56923 C4QSD3 21015140 IC50 = 476 nM T56923 CU79WM 21035680 Ki = 567 nM T56923 CQ2V9Y 21037713 IC50 = 5.7 nM T56923 C1TO9U 21184748 IC50 > 9000 nM T56923 CPJ3A2 21184843 IC50 = 57 nM T56923 CC70HR 21878232 IC50 = 32 nM T56923 C73BVK 21878262 IC50 > 20000 nM T56923 C31CTJ 21878266 IC50 > 20000 nM T56923 C7NFM2 21878293 IC50 > 20000 nM T56923 CC0XY4 21878295 IC50 > 20000 nM T56923 CM7JZ3 21878298 IC50 > 20000 nM T56923 CB3L1Z 21878309 IC50 = 460 nM T56923 CAF9C8 21878315 IC50 > 20000 nM T56923 C1NH7B 22238507 IC50 = 28600 nM T56923 CGFK80 22288470 IC50 = 1000 nM T56923 C9J8CR 22648972 IC50 = 50 nM T56923 CU2BO5 22648978 IC50 = 7000 nM T56923 CE6WA0 22649035 IC50 = 79.43 nM T56923 CPH92E 22649099 IC50 = 31.62 nM T56923 CPJE60 23519822 IC50 = 12.59 nM T56923 C8YM6P 23519825 IC50 = 12.59 nM T56923 CI2K1T 23519852 IC50 = 2 nM T56923 CGM3N9 23709380 IC50 = 0.1 nM T56923 C4Q6RG 24804051 IC50 = 330 nM T56923 CM8BS1 24879232 IC50 = 5 nM T56923 CF9J4A 24952757 IC50 = 810 nM T56923 CT1PY9 24952761 IC50 = 4100 nM T56923 CJF74H 24953110 IC50 = 280 nM T56923 C71SYH 24953463 IC50 = 150 nM T56923 CQ71HO 24953464 IC50 = 260 nM T56923 CW80DI 24953816 IC50 = 870 nM T56923 C0X8AV 24958572 IC50 = 1500 nM T56923 CZX9A5 24958574 IC50 = 910 nM T56923 CTCG15 24958934 IC50 = 470 nM T56923 CW8E4I 24958935 IC50 = 850 nM T56923 CN2ZH9 24958936 IC50 = 510 nM T56923 CU41QF 24958937 IC50 = 820 nM T56923 CE80JT 24958938 IC50 = 1700 nM T56923 C4E9IS 24959296 IC50 = 1700 nM T56923 CK71AE 24959664 IC50 = 4800 nM T56923 CU2Y7H 24959665 IC50 = 6400 nM T56923 C50KTE 24959666 IC50 = 7800 nM T56923 C3IJL1 24959669 IC50 = 4100 nM T56923 C6L0RD 24960030 IC50 = 4100 nM T56923 C5F6RV 25022517 Ki = 2.8 nM T56923 CJ9E8V 25110787 IC50 = 2 nM T56923 C0PIM7 42642630 Ki = 2 nM T56923 CKQ82X 44157035 Ki = 5 nM T56923 CGAU73 44249793 Ki = 4 nM T56923 C1LCP6 44249825 Ki = 4.5 nM T56923 C5YFB9 44252324 IC50 > 10000 nM T56923 COM8G0 44318535 IC50 < 4600 nM T56923 CK23IC 44318556 IC50 = 170 nM T56923 C2I5PW 44318557 IC50 = 300 nM T56923 CS1B2C 44318669 IC50 = 730 nM T56923 CTS6P1 44318749 IC50 = 10000 nM T56923 C62GTK 44318765 IC50 = 92 nM T56923 C3N0JT 44318777 IC50 = 4200 nM T56923 CLO0M1 44318869 IC50 = 4400 nM T56923 CD3H7M 44318872 IC50 = 830 nM T56923 CLK01X 44318921 IC50 = 2800 nM T56923 CF64GM 44393541 IC50 = 10 nM T56923 CGJE30 44393543 IC50 = 114 nM T56923 CRI97S 44393573 IC50 = 906 nM T56923 CSMX21 44407551 IC50 = 3900 nM T56923 CGJD54 44407558 IC50 = 10000 nM T56923 C3B2FZ 44407698 IC50 = 1400 nM T56923 CVCY30 44407774 IC50 = 9.5 nM T56923 C83HJX 44407789 IC50 = 350 nM T56923 C92IWD 44410818 Ki = 600 nM T56923 C3I8QR 44410826 Ki > 5000 nM T56923 CZ59WM 44410827 Ki = 750 nM T56923 CN65UT 44410828 Ki = 57 nM T56923 CS07ZG 44410831 Ki > 10000 nM T56923 CEN90F 44410835 Ki = 85 nM T56923 CR5H6A 44410836 Ki = 100 nM T56923 CNM0S1 44410837 Ki = 43 nM T56923 CD04KH 44410839 Ki = 160 nM T56923 C21KQP 44410842 Ki = 40 nM T56923 CS82VJ 44410894 Ki = 200 nM T56923 CB3J7K 44410898 Ki = 60 nM T56923 C4VNU2 44410899 Ki = 120 nM T56923 CT79SM 44410901 Ki = 290 nM T56923 CDHU68 44410903 Ki = 42 nM T56923 C25XDZ 44410909 Ki = 32 nM T56923 CAC7H2 44410911 Ki = 35 nM T56923 C62RDM 44410912 Ki = 50 nM T56923 CV5TD2 44410937 Ki = 1700 nM T56923 C1WK0C 44410939 Ki = 6000 nM T56923 CG8N6C 44410940 Ki > 10000 nM T56923 C3Q9FW 44410941 Ki = 17 nM T56923 C1JM5T 44410943 Ki = 90 nM T56923 C3JSQ8 44410945 Ki = 27 nM T56923 C6RI4S 44410946 Ki = 37 nM T56923 CT8XZ7 44410952 Ki = 14 nM T56923 CB32PT 44414037 IC50 = 3100 nM T56923 CP0V4L 44414038 IC50 = 1000 nM T56923 CC4O9L 44414052 IC50 = 53 nM T56923 C37XKY 44414053 IC50 = 34 nM T56923 C64LVB 44414071 IC50 = 22 nM T56923 CA75IR 44414095 IC50 = 8600 nM T56923 CZKS05 44414222 IC50 = 548 nM T56923 CI2O0M 44414231 IC50 = 65 nM T56923 CG7V4R 44414232 IC50 = 14 nM T56923 CX0S1E 44414247 IC50 = 139 nM T56923 CXMU80 44414248 IC50 = 41 nM T56923 CL2M8C 44414249 IC50 = 926 nM T56923 C05YEA 44414261 IC50 = 7200 nM T56923 C5LMX2 44414294 IC50 = 56 nM T56923 CLN4R1 44414295 IC50 = 74 nM T56923 CCMI24 44419411 IC50 = 15 nM T56923 C39AZS 44419412 IC50 = 112 nM T56923 CN1WA4 44419439 IC50 = 17 nM T56923 CKID29 44419441 IC50 = 9 nM T56923 C60WDB 44419448 IC50 = 9 nM T56923 C3SAK6 44419449 IC50 = 13 nM T56923 CYBP92 44419473 IC50 = 9 nM T56923 CGT14K 44419476 IC50 = 17 nM T56923 CU3D9L 44419477 IC50 = 7 nM T56923 C7Q2DF 44419479 IC50 = 6 nM T56923 CCS0Q9 44419480 IC50 = 4 nM T56923 CCHS37 44419482 IC50 = 7 nM T56923 CZQ7F9 44419483 IC50 = 12 nM T56923 CXYP53 44419546 IC50 = 12 nM T56923 C1T3XJ 44419555 IC50 = 16 nM T56923 CA4IH6 44419558 IC50 = 22 nM T56923 CE8B9Y 44431171 IC50 = 15.85 nM T56923 CGBC76 44431175 IC50 = 63.1 nM T56923 C93BIU 44431178 IC50 < 1000 nM T56923 C9MQ8S 44431182 IC50 = 19.95 nM T56923 COD27M 44431186 IC50 = 100 nM T56923 C4ZFV1 44431189 IC50 = 31.62 nM T56923 C16IRE 44431193 IC50 = 100 nM T56923 CH70AY 44431195 IC50 = 7.943 nM T56923 C4TSW3 44431196 IC50 = 398.11 nM T56923 CF19NE 44431198 IC50 = 1584.89 nM T56923 C1B6YU 44431207 IC50 = 15.85 nM T56923 CW01YN 44431208 IC50 = 31.62 nM T56923 C4RT3H 44431209 IC50 = 3 nM T56923 C9I5AK 44431210 IC50 = 15.85 nM T56923 C1M6WF 44431211 IC50 = 35 nM T56923 CG85RQ 44432384 IC50 = 2400 nM T56923 C7C6UQ 44432385 IC50 = 740 nM T56923 CAMQ76 44432386 IC50 = 400 nM T56923 C0N8KE 44432388 IC50 = 6100 nM T56923 CGIA14 44432390 IC50 = 5100 nM T56923 C3C0JF 44432391 IC50 = 460 nM T56923 C15MFH 44432392 IC50 = 120 nM T56923 C5S3NL 44432393 IC50 = 3900 nM T56923 CFCO09 44432394 IC50 = 1600 nM T56923 CB7OM5 44432396 IC50 = 390 nM T56923 C3W6AG 44432397 IC50 = 230 nM T56923 C51DUO 44432415 IC50 = 250 nM T56923 CB6J0H 44432416 IC50 = 54 nM T56923 C7J1KU 44432417 IC50 = 830 nM T56923 CJH41P 44432418 IC50 = 930 nM T56923 CX0O3H 44432419 IC50 > 30000 nM T56923 C5FXB7 44432420 IC50 = 4500 nM T56923 C7CN1J 44432421 IC50 > 30000 nM T56923 CQM21O 44432422 IC50 = 360 nM T56923 CBO05K 44432423 IC50 = 70 nM T56923 CBA86X 44432435 IC50 = 280 nM T56923 C32JQN 44432436 IC50 = 3000 nM T56923 C6MO0Y 44432437 IC50 = 480 nM T56923 CFA91Q 44439676 IC50 = 205 nM T56923 C6HG8Y 44439677 IC50 = 52 nM T56923 CH0RY4 44439678 IC50 = 308 nM T56923 C5B6XJ 44439680 IC50 = 54 nM T56923 C9QA2V 44439682 IC50 = 1720 nM T56923 CMD0L2 44439685 IC50 = 358 nM T56923 C4I7NW 44439699 IC50 > 30000 nM T56923 CB50CX 44439700 IC50 > 30000 nM T56923 CEY17F 44439701 IC50 = 15 nM T56923 C6X4CH 44439702 IC50 = 8 nM T56923 C0D1JK 44439704 IC50 = 13 nM T56923 CHJ4G3 44439706 IC50 = 8 nM T56923 CH15WA 44439708 IC50 = 10 nM T56923 CI7XA6 44439720 IC50 = 28 nM T56923 CY2I5W 44439723 IC50 = 27 nM T56923 COCV10 44439728 IC50 = 44 nM T56923 CY1B2H 44440858 Ki = 5 nM T56923 CN4ZL9 44440859 Ki = 10 nM T56923 CN90ZV 44440860 Ki = 25 nM T56923 C0GZB2 44440865 Ki = 0.6 nM T56923 CG01PI 44440866 Ki = 0.8 nM T56923 CC1Z2N 44440873 Ki = 4 nM T56923 C07WNS 44446565 IC50 = 4.1 nM T56923 CALE50 44446566 IC50 = 4.7 nM T56923 C9OW0Z 44446567 IC50 = 4.8 nM T56923 CGM98S 44446568 IC50 = 17.2 nM T56923 CXJ51G 44446569 IC50 = 6.8 nM T56923 C9DCO6 44446570 IC50 = 2.8 nM T56923 C5EY8W 44446571 IC50 = 94 nM T56923 C15IZA 44446572 IC50 = 171 nM T56923 C34XTN 44446577 IC50 = 49 nM T56923 C3ZU9O 44446578 IC50 = 150 nM T56923 CW63PF 44446580 IC50 = 58 nM T56923 C5QWB7 44446583 IC50 = 87 nM T56923 CJZ13N 44446593 IC50 = 4.5 nM T56923 CEK28S 44446595 IC50 = 5 nM T56923 C7VE2J 44446596 IC50 = 6.1 nM T56923 C71OQP 44446598 IC50 = 9.5 nM T56923 CPK8T3 44446602 IC50 = 8.2 nM T56923 C5CAE9 44446604 IC50 = 7.6 nM T56923 CA0K6E 44446605 IC50 = 16.5 nM T56923 C3TZV2 44446607 IC50 = 8.6 nM T56923 C31JGN 44446608 IC50 = 10.9 nM T56923 C9R2IX 44446610 IC50 = 9.8 nM T56923 C91YQW 44446611 IC50 = 9.8 nM T56923 CBLF23 44446613 IC50 = 7.5 nM T56923 C1N9QM 44446614 IC50 = 8.2 nM T56923 C54CVM 44446616 IC50 = 8 nM T56923 CB2VC0 44446617 IC50 = 5.8 nM T56923 C8OUJ2 44446621 IC50 = 6.2 nM T56923 C6AGR1 44446631 IC50 = 21 nM T56923 CO2C6K 44446633 IC50 = 815 nM T56923 CTF63M 44446635 IC50 = 50 nM T56923 CKGN35 44446639 IC50 = 4.6 nM T56923 CIDA76 44446641 IC50 = 3.8 nM T56923 CZ7S4Y 44446645 IC50 = 6.3 nM T56923 CTO73Z 44446647 IC50 = 3.4 nM T56923 CEZ48V 44446650 IC50 = 3.3 nM T56923 CON0S6 44447608 IC50 = 3.5 nM T56923 CSXY76 44447915 IC50 = 72 nM T56923 C7SO8Z 44447916 IC50 > 2000 nM T56923 CT10JA 44447917 IC50 = 170 nM T56923 CYR3D8 44447918 IC50 = 64 nM T56923 CAYO93 44447919 IC50 = 1300 nM T56923 CSO28V 44447920 IC50 = 1400 nM T56923 CHF86G 44447921 IC50 = 220 nM T56923 CPD90B 44447922 IC50 = 260 nM T56923 CP3R7Q 44447923 IC50 = 70 nM T56923 C28JNX 44447924 IC50 = 160 nM T56923 CR6N4Y 44447925 IC50 = 19 nM T56923 CT29LR 44447928 IC50 = 14 nM T56923 CR31IU 44447929 IC50 = 66 nM T56923 CZ61DE 44447931 IC50 = 1100 nM T56923 CU4QD0 44447932 IC50 = 1100 nM T56923 CU87FV 44447933 IC50 = 880 nM T56923 CD64WU 44447937 IC50 = 260 nM T56923 CB58DL 44447939 IC50 = 150 nM T56923 CF7X8N 44447942 IC50 = 57 nM T56923 C6NM4J 44447943 IC50 = 24 nM T56923 C4LO0R 44447944 IC50 = 90 nM T56923 C80PWE 44447945 IC50 = 640 nM T56923 CL90IY 44447946 IC50 = 4 nM T56923 CZ6LD3 44447947 IC50 = 400 nM T56923 CPN94Y 44447948 IC50 = 520 nM T56923 C6OPD7 44447949 IC50 = 140 nM T56923 CA8EC9 44447950 Ki = 28 nM T56923 CWZ6F9 44447951 Ki = 5.2 nM T56923 C9OG3A 44447952 Ki = 1.5 nM T56923 C87MKS 44447953 Ki = 19.4 nM T56923 CT7S3K 44447954 Ki = 13.9 nM T56923 CTU25R 44447955 Ki = 6.1 nM T56923 C46ZLO 44447956 Ki = 11.9 nM T56923 C4AB2Z 44447957 Ki = 16 nM T56923 CZ0I9N 44447958 Ki = 38.5 nM T56923 CC34NQ 44447959 Ki = 1.7 nM T56923 CHWV97 44447960 Ki = 1.9 nM T56923 CQ10GH 44447961 Ki = 4.5 nM T56923 C4UR8M 44447962 Ki = 7.9 nM T56923 CRE30Q 44447963 Ki = 13.3 nM T56923 C8AZ7N 44447964 Ki = 11.8 nM T56923 CR17NJ 44447965 Ki = 4.4 nM T56923 CLWV47 44447966 Ki = 1 nM T56923 CJN4H6 44447967 Ki = 1.9 nM T56923 C1GY9W 44447968 Ki = 1.7 nM T56923 CI5D9J 44454958 IC50 = 2500 nM T56923 CZI7F6 44454985 IC50 = 2 nM T56923 CI3S2D 44454986 IC50 = 45 nM T56923 C4OVB0 44455010 IC50 = 16 nM T56923 CY0KX8 44455012 IC50 = 350 nM T56923 CY54PX 44455014 IC50 = 1 nM T56923 CJ2DF1 44455045 IC50 = 5 nM T56923 CPI2L7 44455083 IC50 = 280 nM T56923 C82AZU 44455116 IC50 = 280 nM T56923 C8D3GL 44455117 IC50 = 140 nM T56923 C7QHN1 44455191 IC50 = 630 nM T56923 CKO9T3 44455234 IC50 = 13 nM T56923 CVA0H4 44455386 IC50 = 60 nM T56923 C3S4NC 44455404 IC50 = 5 nM T56923 C4DL5C 44469677 IC50 > 10000 nM T56923 C8ZLV4 44564898 Ki = 5 nM T56923 CD6EW2 44564940 Ki = 400 nM T56923 C2NFZ7 44564941 Ki = 13 nM T56923 C43RSH 44564942 Ki = 4 nM T56923 CO1WZ3 44564943 Ki = 7 nM T56923 C2U9OC 44564998 Ki = 12 nM T56923 CAK9P0 44564999 Ki = 2 nM T56923 C28OAW 44565049 Ki = 5 nM T56923 CW3G1V 44565050 Ki = 9 nM T56923 C76YJU 44565051 Ki = 8 nM T56923 CP1RO6 44565052 Ki = 4 nM T56923 CG4I0V 44565098 Ki = 7 nM T56923 CHX49N 44565099 Ki = 5 nM T56923 C3LAO8 44565100 Ki = 5 nM T56923 CH8FP0 44565148 Ki = 14 nM T56923 CN8PI3 44610601 IC50 = 2 nM T56923 C8HD1U 44626319 IC50 = 0.12 nM T56923 C10RHQ 44775716 IC50 = 390 nM T56923 CQF5V1 45268603 Ki = 12 nM T56923 CMF07V 45269458 Ki > 270 nM T56923 CZ84AK 45269459 Ki > 270 nM T56923 CN8S4C 45270317 Ki > 2000 nM T56923 CQF0A4 45271150 Ki = 5 nM T56923 CTX49I 45271151 Ki = 50 nM T56923 CZI5C3 45272016 Ki = 22 nM T56923 C4DVZ5 45272017 Ki > 270 nM T56923 CM8PG5 45272018 Ki > 270 nM T56923 C3QO9B 45272020 Ki = 34 nM T56923 CIMJ26 45272042 Ki = 15 nM T56923 CM2BA6 45272064 Ki = 76 nM T56923 C0QZT7 45272839 Ki = 219 nM T56923 C9NR1T 45272847 Ki = 5 nM T56923 CI51QN 45272856 Ki = 203 nM T56923 CDB27G 45272863 Ki = 17 nM T56923 CNXJ43 45272873 Ki = 61 nM T56923 CLF16N 45485721 IC50 = 5490 nM T56923 CSP9M7 45485756 Ki = 320 nM T56923 C3EL4C 45485757 IC50 = 54 nM T56923 C7J8IO 45485758 Ki = 550 nM T56923 CX6ZG2 45485775 IC50 = 100 nM T56923 CKU6S2 45485784 IC50 = 75 nM T56923 CV48KD 45485788 IC50 = 6340 nM T56923 CUE8N7 45485798 Ki = 260 nM T56923 CK3N1G 46206137 IC50 > 10000 nM T56923 CYKF43 46896583 IC50 > 5000 nM T56923 CLM9W0 46896584 IC50 > 10000 nM T56923 C6PZT7 46896587 IC50 > 5000 nM T56923 C97LJK 46896679 IC50 > 5000 nM T56923 CG40RT 46896680 IC50 = 540 nM T56923 CF4JN7 46896681 IC50 > 5000 nM T56923 CS9N0R 46896682 IC50 > 5000 nM T56923 CJ4U6X 46896684 IC50 > 10000 nM T56923 CV1M9N 46896685 IC50 > 5000 nM T56923 CW7NC4 46896779 IC50 > 10000 nM T56923 C2U7AK 46896780 IC50 > 5000 nM T56923 C6C3NI 46896781 IC50 > 10000 nM T56923 C7LYG6 46896884 IC50 > 10000 nM T56923 C0CEV2 46897163 IC50 = 21 nM T56923 COG3A1 46897256 IC50 = 277 nM T56923 C1AO8D 46897352 IC50 = 275 nM T56923 CD14NQ 46897356 IC50 = 759 nM T56923 CUQ5P1 46897447 IC50 > 5000 nM T56923 C7SQA3 46897448 IC50 > 10000 nM T56923 CD8KM2 46897449 IC50 = 1480 nM T56923 CVLA96 46897450 IC50 = 2120 nM T56923 CX8YD0 46897451 IC50 = 170 nM T56923 CH9B3S 46897452 IC50 = 1610 nM T56923 C72LPT 46897453 IC50 > 10000 nM T56923 CVE23C 46897537 IC50 > 5000 nM T56923 CL0K1O 46897538 IC50 > 10000 nM T56923 C7E8PR 46897539 IC50 > 10000 nM T56923 C6CFK0 46897540 IC50 > 10000 nM T56923 C9ZSC0 46897628 IC50 > 10000 nM T56923 CN7WF3 46897629 IC50 > 10000 nM T56923 CHZ1R4 46897630 IC50 > 5000 nM T56923 C8DMT7 46897631 IC50 > 10000 nM T56923 C16BTL 46897632 IC50 > 5000 nM T56923 C1NJ0H 46897731 IC50 > 10000 nM T56923 CU1PG4 46897732 IC50 > 5000 nM T56923 CAXG02 46897733 IC50 > 5000 nM T56923 CN1A6E 46897734 IC50 > 5000 nM T56923 C6B4YM 46897735 IC50 > 10000 nM T56923 CFR6L3 46897736 IC50 > 5000 nM T56923 CN6B9F 46897737 IC50 > 5000 nM T56923 CKH1N7 49763036 IC50 = 2 nM T56923 C78MYC 56839292 IC50 > 5000 nM T56923 CD35UF 56839293 IC50 > 5000 nM T56923 CTFL56 56839294 IC50 = 1100 nM T56923 CYA2V8 56839499 IC50 = 121 nM T56923 C3Y0XZ 57692074 Ki = 79 nM T56923 CJ6S4P 57833094 IC50 = 7.943 nM T56923 CJ86XP 57833099 IC50 = 79.43 nM T56923 COZ10N 57833129 IC50 = 3162.28 nM T56923 CC3S2Z 57833135 IC50 = 10 nM T56923 CMI3G0 57833157 IC50 = 31.62 nM T56923 C34ROA 57833159 IC50 = 79.43 nM T56923 CQ9I7S 57833164 IC50 = 50.12 nM T56923 CMV0U6 57833185 IC50 = 5.012 nM T56923 CV4QX5 57833195 IC50 = 63.1 nM T56923 C8DR7C 57833197 IC50 = 398.11 nM T56923 C4B0TK 57833198 IC50 = 31.62 nM T56923 C86YSD 57833203 IC50 = 158.49 nM T56923 CU3W6L 57833212 IC50 = 31.62 nM T56923 C6ZF0T 57833215 IC50 = 158.49 nM T56923 CS58RL 58180198 IC50 = 0.3162 nM T56923 CUFZ86 58180199 IC50 = 0.3162 nM T56923 C3SX6B 58180205 IC50 = 0.3162 nM T56923 CUZ3B8 58230405 Ki = 530 nM T56923 C9HBX4 58230406 Ki = 1980 nM T56923 CXJW13 58230407 Ki = 1790 nM T56923 C0YWT1 58509213 IC50 > 10000 nM T56923 CJ3CE7 59446379 IC50 > 10000 nM T56923 C7G1XO 59446380 IC50 = 1990 nM T56923 C7S2LF 59446381 IC50 = 278 nM T56923 CH69IX 59446384 IC50 = 78 nM T56923 C9C7MA 59446394 IC50 > 10000 nM T56923 C7NOM4 59446412 IC50 = 3900 nM T56923 CW4SR2 59799570 Ki = 510 nM T56923 C2GQ8H 66622526 Ki = 920 nM T56923 C8WC7S 66856548 IC50 = 1100 nM T56923 CK01EX 68084172 IC50 = 25.12 nM T56923 CI19WL 68603807 IC50 = 1700 nM T56923 CFH79W 69440865 Ki = 4.1 nM T56923 C2C4RW 69441619 Ki = 580 nM T56923 CX7W5R 69442228 Ki = 460 nM T56923 CV86DX 71624890 Ki = 100 nM T56923 CE0GS7 71625019 Ki = 4200 nM T56923 C6B8IX 71625020 Ki = 1940 nM T56923 CPD5U8 71625021 Ki = 2400 nM T56923 CQ70HI 71625022 Ki = 5900 nM T56923 CR4C3X 71625144 Ki = 150 nM T56923 CDC34R 71625146 Ki = 370 nM T56923 CK4J5A 71625271 Ki = 1750 nM T56923 C0U6DF 71625272 Ki = 220 nM T56923 C0A6VG 71625273 Ki = 1500 nM T56923 CM6KB1 71625274 Ki = 4100 nM T56923 CXHS27 71625275 Ki = 590 nM T56923 C43XWU 71625276 Ki = 190 nM T56923 C3EG4B 71625389 Ki = 1600 nM T56923 CY2RQ6 71625390 Ki = 258 nM T56923 CP4QS0 71625391 Ki = 79 nM T56923 C6CW4Y 71625392 Ki = 64 nM T56923 CN83DJ 71625501 Ki = 5400 nM T56923 C7S0CI 71625502 Ki = 9000 nM T56923 CQ2Z3N 71625503 Ki = 349 nM T56923 C9N4FO 71625504 Ki = 523 nM T56923 C7Q2FV 71625505 Ki = 2600 nM T56923 C2GKN5 71625506 Ki = 6000 nM T56923 CP9E7K 71625625 Ki = 13000 nM T56923 CI0GU8 71660496 IC50 > 48500 nM T56923 C1N4GD 71716556 Ki = 1129 nM T56923 CA89MZ 71718998 Ki = 489 nM T56923 C7RUD1 71720196 Ki = 220 nM T56923 CWH6T3 72548703 IC50 = 0.24 nM T56923 C8L4CY 72947875 IC50 > 30000 nM T56923 CLJN23 72947876 IC50 > 30000 nM T56923 CMP17R 72947877 IC50 = 11000 nM T56923 C2TZQ4 72947878 IC50 = 13000 nM T56923 C7BVT2 72948068 IC50 = 11000 nM T56923 CT3WY8 72948071 IC50 = 20000 nM T56923 C9W1XN 72948072 IC50 = 10500 nM T56923 CLAY08 72948073 IC50 = 13900 nM T56923 C8EN0I 77844166 IC50 > 5000 nM T56923 C5IP8A 90292839 IC50 > 5000 nM T56923 C3XR4O 91937330 IC50 = 520 nM T56923 C38FJW 91937331 IC50 = 105 nM T56923 C9Y4MA 91937332 IC50 = 294 nM T56923 C48LAC 91937333 IC50 = 890 nM T56923 C6ENV5 100951623 IC50 = 5.2 nM T56923 C07RBY 101885088 IC50 > 10000 nM T56923 C2DS5Y 118540482 IC50 = 1 nM T56923 CWN5E2 118540525 IC50 = 1 nM T56923 CXY73S 118540528 IC50 = 1.259 nM T56923 C0B5EO 118540567 IC50 = 1 nM T56923 C25VOY 118540730 IC50 = 0.3981 nM T56923 C0QP7G 118540796 IC50 = 1.585 nM T56923 CCB30T 118540867 IC50 = 0.2512 nM T56923 CE01XS 118540892 IC50 = 0.1995 nM T56923 CPW24Q 118554742 IC50 = 0.5012 nM T56923 CHB78C 118554743 IC50 = 0.2512 nM T56923 C9H2XV 118554752 IC50 = 31.62 nM T56923 CE1K8F 118554754 IC50 = 0.7943 nM T56923 CE8R9Q 118554755 IC50 = 1.259 nM T56923 CBLI90 118554787 IC50 = 0.631 nM T56923 C12GOL 118554789 IC50 = 2.512 nM T56923 CI1JV8 118554794 IC50 = 0.5012 nM T56923 C3U6XS 118554808 IC50 = 316.23 nM T56923 CL7Y5T 118554809 IC50 = 0.5012 nM T56923 C0Z9PG 118554832 IC50 = 0.1995 nM T56923 C1ELW7 118554833 IC50 = 316.23 nM T56923 C41OZF 118554834 IC50 = 1 nM T56923 CR18SU 118554836 IC50 = 1 nM T56923 CV8BD0 118554882 IC50 = 0.5012 nM T56923 C4SVK9 118706787 IC50 > 30000 nM T56923 CH2S7P 118706788 IC50 > 30000 nM T56923 CEO2D1 118716381 IC50 > 10000 nM T56923 C8Z0HW 118720448 IC50 > 10000 nM T56923 CS58IW 118730035 IC50 = 398.11 nM T56923 CDEQ15 118730036 IC50 = 794.33 nM T56923 CY0TC4 118730037 IC50 = 7943.28 nM T56923 C02COA 118730038 IC50 = 630.96 nM T56923 C8I7HQ 118730039 IC50 > 10000 nM T56923 C3YNJ7 122187254 IC50 = 733 nM T56923 CUL9I1 122187255 IC50 = 410 nM T56923 CCD97V 122187256 IC50 = 2200 nM T56923 C6MW4Q 122187257 IC50 = 81 nM T56923 CUFD82 122187258 IC50 > 5000 nM T56923 CHNY79 122187259 IC50 = 918 nM T56923 C6HB2K 122187260 IC50 = 2500 nM T56923 CQ16CH 122187261 IC50 = 2600 nM T56923 CD7Z4N 122187262 IC50 = 933 nM T56923 C9V7XK 122187263 IC50 = 298 nM T56923 CE8S4F 122187264 IC50 = 4850 nM T56923 CO5UZ9 122187265 IC50 = 2300 nM T56923 CEZ14H 122187266 IC50 = 21 nM T56923 CRBQ58 122187267 IC50 > 5000 nM T56923 C0VD5A 122187268 IC50 = 4 nM T56923 CQB0L1 122187269 IC50 = 4310 nM T56923 CY1S7I 122187270 IC50 > 5000 nM T56923 CF89ON 122187271 IC50 = 655 nM T56923 C6B5NM 123159150 IC50 = 3.162 nM T56923 CIY58P 123190913 IC50 = 0.3981 nM T56923 CR4XJ8 123227682 IC50 = 10 nM T56923 CIY85P 123626575 IC50 = 25.12 nM T56923 CS1B2E 127020968 IC50 = 25.12 nM T56923 C85ULI 127048710 IC50 = 7.943 nM T56923 CZV7Q0 127049047 IC50 = 1.585 nM T56923 CB54VQ 127049048 IC50 = 158.49 nM T56923 C9TUQ2 127049049 IC50 = 1.259 nM T56923 CW3Q9B 127049108 IC50 = 1 nM T56923 C6LI9P 127049370 IC50 = 0.5012 nM T56923 C59WMS 127049371 IC50 = 100 nM T56923 CS3Q0P 127049422 IC50 = 0.7943 nM T56923 C6WC3F 127049427 IC50 = 1.585 nM T56923 CF76RT 127049428 IC50 = 3162.28 nM T56923 C27QHU 127049429 IC50 = 10 nM T56923 C4KMR9 127049430 IC50 = 6309.57 nM T56923 CK2AO1 127049431 IC50 = 0.3981 nM T56923 C67ZBO 127049432 IC50 = 0.631 nM T56923 C8MVR5 127050016 IC50 = 0.7943 nM T56923 CS34YB 127050017 IC50 = 1.995 nM T56923 COTZ42 127050964 IC50 = 0.5012 nM T56923 CS7W3P 127051212 IC50 = 0.5012 nM T56923 C1TY2F 127051854 IC50 = 0.3981 nM T56923 CGY3S7 127052172 IC50 = 1.995 nM T56923 CROV30 127052173 IC50 = 0.3981 nM T56923 CQ19WY 127052174 IC50 = 7.943 nM T56923 C3TCM5 129315964 IC50 = 0.631 nM T56923 C3ZFT2 129315976 IC50 = 2511.89 nM T56923 CVAY21 129315983 IC50 = 1.259 nM T56923 C98MZR 129315994 IC50 = 3.981 nM T56923 C3EXG0 129315999 IC50 = 1.585 nM T56923 C06ZVX 129316000 IC50 = 3.981 nM T56923 COS96P 129316018 IC50 = 0.3981 nM T56923 COA51I 129316022 IC50 = 6.31 nM T56923 C7FG4C 129316023 IC50 = 79.43 nM T56923 C6FYS9 129316027 IC50 = 1.995 nM T56923 C86EAY 129316028 IC50 = 0.3162 nM T56923 CY16MX 129316030 IC50 = 100 nM T56923 CL9SY6 129316051 IC50 = 125.89 nM T56923 CZ4R0O 129316053 IC50 = 1.259 nM T56923 CQ85LF 129316058 IC50 = 501.19 nM T56923 CG90CF 129316069 IC50 = 0.2512 nM T56923 C2OHC7 129316073 IC50 = 251.19 nM T56923 CHM7P9 129316076 IC50 = 1.995 nM T56923 CX5W0K 130191301 IC50 = 1 nM T56923 CR81QZ 135286501 IC50 = 17 nM T56923 CBJ90L 135405057 Ki = 4.7 nM T56923 CL9BV0 135497124 IC50 = 21 nM T56923 CGJ8I4 135508400 IC50 = 20000 nM T56923 CEHP65 135531169 IC50 = 270 nM T56923 CA45JR 135534060 IC50 = 4300 nM T56923 C9XUH4 135539055 Ki = 11 nM T56923 CVLK72 135555955 IC50 = 1300 nM T56923 C6J7ZP 135673987 IC50 = 10000 nM T56923 CEL95R 135673991 IC50 = 480 nM T56923 C2RDY4 135814570 Ki = 5110 nM T56923 CT2UB0 135907759 IC50 = 710 nM T56923 C57BCE 135907763 IC50 = 780 nM T56923 CB9IT0 135907764 IC50 = 140 nM T56923 C39AME 135907765 IC50 = 3700 nM T56923 COXZ12 135907766 IC50 = 7400 nM T56923 C9N8JV 135907767 IC50 = 1400 nM T56923 CN29YM 135907772 IC50 = 4700 nM T56923 C3BS2U 135907774 IC50 = 1600 nM T56923 C6XMV7 135907779 IC50 = 4900 nM T56923 CT1K4R 135907780 IC50 = 4600 nM T56923 C0Y8AW 135907781 IC50 = 1700 nM T56923 C4GP2U 135907782 IC50 = 900 nM T56923 C86LGZ 135907789 IC50 = 3700 nM T56923 CZ0M8U 135907792 IC50 = 4300 nM T56923 C16YJA 135907804 IC50 = 10 nM T56923 C8X7UT 135937901 Ki = 330 nM T56923 C5GY0S 135949064 IC50 = 6 nM T56923 C8NO4C 135950089 IC50 = 8000 nM T56923 C50YXB 135950090 IC50 > 30000 nM T56923 CMA1E9 135964204 IC50 = 510 nM T56923 CID30V 136036234 Ki = 10000 nM T56923 CI4PS1 136036235 Ki = 1300 nM T56923 C7FX0N 136036236 Ki = 3000 nM T56923 C1NF6Y 136036238 Ki = 2280 nM T56923 CH78DC 136036240 Ki = 10000 nM T56923 C0YVI5 136036241 IC50 = 36 nM T56923 CME5L2 136036242 Ki = 381 nM T56923 CQ2VE9 136036243 Ki = 2360 nM T56923 C5AR1O 136036244 Ki = 1300 nM T56923 CRN73I 136036245 Ki = 1270 nM T56923 CSL40I 136036246 Ki = 749 nM T56923 C3ZUN6 136036249 Ki = 168 nM T56923 COB78Q 136036250 Ki = 114 nM T56923 C2CO6U 136036251 Ki = 79 nM T56923 CNV4H2 136036252 Ki = 44 nM T56923 CA8JF5 136036253 Ki = 10000 nM T56923 CR8LO7 136036254 Ki = 4300 nM T56923 C6O0PW 136036255 Ki = 4100 nM T56923 CI2L5T 136036256 Ki = 2030 nM T56923 C6FS8C 136036257 Ki = 10000 nM T56923 CXZ4F3 136036517 Ki = 24 nM T56923 CLF7E4 136036518 Ki = 9 nM T56923 C4FRC5 136036519 Ki = 11 nM T56923 C67PHR 136036520 Ki = 184 nM T56923 CSK0N6 136036521 Ki = 16 nM T56923 CU4YJ8 136036522 Ki = 9 nM T56923 CFYG04 136060643 IC50 = 15000 nM T56923 C08WRM 136074340 IC50 = 1300 nM T56923 CZ71YS 136074341 IC50 = 7 nM T56923 CI68DK 136074342 IC50 = 4800 nM T56923 C8BF6W 136074343 IC50 = 6400 nM T56923 C2PQ7L 136074344 IC50 > 30000 nM T56923 C6CL9A 136074345 IC50 = 10000 nM T56923 CSC5H6 136087068 IC50 = 630.96 nM T56923 C9XV7O 136087069 IC50 = 501.19 nM T56923 CO2XD8 136087070 IC50 = 316.23 nM T56923 CU6SF2 136087071 IC50 = 2511.89 nM T56923 CQ27TY 136087072 IC50 = 630.96 nM T56923 CQJE63 136087073 IC50 = 630.96 nM T56923 C7J4GD 136087074 IC50 = 2511.89 nM T56923 C08HGI 136087075 IC50 = 2511.89 nM T56923 CY7D1S 136087076 IC50 = 398.11 nM T56923 C3MIC4 136087077 IC50 > 10000 nM T56923 CS0OP1 136087078 IC50 = 251.19 nM T56923 CWS53V 136087079 IC50 = 199.53 nM T56923 CW5Q0X 136087080 IC50 = 125.89 nM T56923 C07RVQ 136087081 IC50 = 6.31 nM T56923 CT7PR1 136087082 IC50 = 398.11 nM T56923 CG69XD 136087083 IC50 = 15.85 nM T56923 C5SPR1 136087084 IC50 = 19.95 nM T56923 CXY58R 136087085 IC50 = 31.62 nM T56923 CB0MG7 136087086 IC50 = 15.85 nM T56923 CM6IR8 136087087 IC50 = 125.89 nM T56923 CUX42V 136087088 IC50 = 100 nM T56923 C58PSH 136087089 IC50 = 125.89 nM T56923 C3O2JS 136087090 IC50 = 630.96 nM T56923 C2I3ZA 136087091 IC50 = 2511.89 nM T56923 C52WRM 136087092 IC50 > 10000 nM T56923 CP9S5K 136087093 IC50 = 25.12 nM T56923 C39WUZ 136087094 IC50 = 50.12 nM T56923 CA40QH 136087095 IC50 = 251.19 nM T56923 C6AB8K 136087096 IC50 = 630.96 nM T56923 CT7WQ9 136986968 IC50 = 320 nM T56923 CUG8T7 136986993 IC50 = 1400 nM T56923 C3IJ0P 136986994 IC50 = 3200 nM T56923 CA46PB 137633482 IC50 = 10 nM T56923 CIT4C2 137633598 IC50 = 0.1585 nM T56923 C7STU9 137634452 IC50 = 25.12 nM T56923 CVJA17 137636599 IC50 > 10000 nM T56923 C3BHQ9 137637097 IC50 = 12.59 nM T56923 C0BF6K 137638965 IC50 = 10 nM T56923 C6SM5N 137639152 IC50 = 158.49 nM T56923 CMWF52 137644193 IC50 = 1258.93 nM T56923 CTK32S 137644508 IC50 = 10 nM T56923 CST9R5 137645182 IC50 = 199.53 nM T56923 C8Q3BK 137645186 IC50 = 1584.89 nM T56923 C1E5HP 137646150 IC50 = 39.81 nM T56923 C91OCN 137649241 IC50 > 10000 nM T56923 CFYA79 137650877 IC50 = 630.96 nM T56923 CC9V4K 137651658 IC50 = 50.12 nM T56923 C1RB2C 137653746 IC50 = 251.19 nM T56923 CX3Z7U 137654230 IC50 = 10 nM T56923 C8YE6L 137657195 IC50 = 316.23 nM T56923 CQV10J 137662215 IC50 = 63.1 nM T56923 CTN2K7 151755055 IC50 = 14800 nM T56923 CAF2H5 155531736 IC50 = 48 nM T56923 C17LKA 155545500 IC50 = 2500 nM T56923 D05AZU 11184341 IC50 = 200 nM T56923 D05CCF 3791448 IC50 = 950 nM T56923 D05SNR 135546485 IC50 = 10000 nM T56923 D06MBD 11176403 IC50 < 3000 nM T56923 D06WVV 11414633 IC50 = 860 nM T56923 D09MAZ 46897162 IC50 = 38 nM T56923 D0D8LQ 9949456 IC50 = 25 nM T56923 D0FF6S 16038374 IC50 > 10000 nM T56923 D0J1XP 11818139 IC50 = 10900 nM T56923 D0T4KC 44439692 IC50 = 276 nM T56923 D0U2UJ 3618472 IC50 = 320 nM T62266 D0B5HS 405012 IC50 = 262700 nM T62266 D0PM5U 135564890 IC50 = 710 nM T62266 CA1H8B 336270 IC50 = 18400 nM T62266 C46VHU 478572 Ki = 5600 nM T62266 C72ZLN 478574 IC50 = 1200 nM T62266 CC7IW3 478577 IC50 = 32000 nM T62266 C2ZR8M 478643 Ki = 13200 nM T62266 CY38AJ 478645 IC50 = 37800 nM T62266 CZT01E 478647 IC50 = 19500 nM T62266 CGT4O9 85469240 Ki = 19860 nM T62266 C8T0MJ 85469241 IC50 = 22220 nM T62266 C5SWD9 85469242 Ki = 45330 nM T62266 CA5CG1 85469243 IC50 = 17760 nM T62266 C5R6WS 85469292 IC50 = 48670 nM T62266 C3Z8YX 91758737 Ki = 6320 nM T62266 CC6VJ5 122525709 Ki = 8850 nM T62266 CY0X9D 122525711 IC50 = 3810 nM T62266 CZE79W 122525712 Ki = 1960 nM T62266 C51WNS 122606362 Ki = 17540 nM T62266 CGO29F 122608329 Ki = 6110 nM T62266 CWDH25 155511770 IC50 = 590 nM T62266 C4H8XB 155536067 IC50 = 280 nM T62266 CFKI70 155539267 IC50 = 490 nM T62266 CH96DK 155550037 IC50 = 25000 nM T62266 CBYL12 155559016 IC50 = 32000 nM T62266 C5Z8YM 155565919 IC50 = 20320 nM T62266 D01HST 1085108 IC50 > 250000 nM T62266 D06YFT 676159 IC50 = 35000 nM T62266 D0I9AT 73549 IC50 = 5000 nM T62266 D0Z3NE 478573 Ki = 970 nM T71230 D03VNJ 16129708 EC50 = 0.1 nM T71230 C0EDH1 44301581 Ki = 62 nM T71230 C4T0MB 44301645 Ki = 680 nM T71230 C8M2XU 44301646 Ki = 0.3 nM T71230 C9AME2 44301661 Ki > 10 nM T71230 CZ4Y6B 44301714 Ki > 10 nM T71230 CRQ1L0 44301718 Ki = 0.49 nM T71230 C9SZ3D 44301732 Ki = 0.4 nM T71230 C02LJW 44301739 Ki = 65 nM T71230 CE0AU3 44301746 Ki = 2600 nM T71230 CDCM97 44301748 Ki = 2900 nM T71230 C5O3NG 44301749 Ki = 539 nM T71230 CGO6W5 44301973 Ki = 87 nM T71230 CDV2Z1 131717293 IC50 = 120 nM T71230 C23SAC 137632225 EC50 = 10000 nM T71230 CUMV75 137634572 EC50 > 50000 nM T71230 C3QBE8 137635347 EC50 = 720 nM T71230 CUDW36 137636118 EC50 = 1100 nM T71230 CE1IC8 137636347 IC50 > 1000 nM T71230 CJX30M 137636606 IC50 > 1000 nM T71230 C3CA5Q 137636877 IC50 > 1000 nM T71230 CYB18U 137637410 EC50 = 30000 nM T71230 CS9NR3 137637531 EC50 = 5.8 nM T71230 COA5V7 137637572 IC50 > 1000 nM T71230 CLB82Z 137638007 IC50 > 1000 nM T71230 CW3Y4G 137638410 EC50 = 73 nM T71230 C8E2CA 137638504 EC50 = 64000 nM T71230 C19FLA 137639109 IC50 > 1000 nM T71230 CI9P2O 137639689 EC50 > 10000 nM T71230 C85BYF 137640890 EC50 = 170 nM T71230 CKC79W 137640954 IC50 > 1000 nM T71230 CW2F3O 137641759 EC50 = 1400 nM T71230 CF8TO7 137642743 IC50 > 1000 nM T71230 CQEP84 137642780 IC50 > 1000 nM T71230 C9H2IK 137642886 EC50 = 5000 nM T71230 CCS6T3 137643048 EC50 = 8.1 nM T71230 C5HB8U 137643294 EC50 = 0.1 nM T71230 C4DHJ5 137643645 IC50 > 1000 nM T71230 CK6U0S 137645853 IC50 > 1000 nM T71230 CM28IO 137646295 EC50 > 50000 nM T71230 CAZC92 137646317 IC50 > 1000 nM T71230 CK0E4W 137647192 EC50 = 260 nM T71230 CJ2PC6 137648579 IC50 > 1000 nM T71230 CUX6D5 137648699 EC50 = 13000 nM T71230 C4RHT7 137649996 IC50 > 1000 nM T71230 CFV35E 137649998 IC50 > 1000 nM T71230 CRA3C4 137650242 EC50 = 220 nM T71230 CWG42U 137651404 IC50 > 1000 nM T71230 CVY34O 137652046 IC50 > 1000 nM T71230 C2IJ8L 137652352 EC50 = 45000 nM T71230 C47ZKI 137652546 IC50 > 1000 nM T71230 C9SX8O 137653764 EC50 = 3400 nM T71230 C49CYT 137654685 IC50 > 1000 nM T71230 C01HOG 137655156 EC50 = 7900 nM T71230 C56LCP 137655239 EC50 = 13000 nM T71230 CP2BY1 137655577 EC50 = 4000 nM T71230 CX6M5O 137656853 IC50 > 1000 nM T71230 CEC4S2 137657880 IC50 > 1000 nM T71230 CX5JC9 137658383 EC50 = 22000 nM T71230 CWH19J 137659661 IC50 > 1000 nM T71230 C0OAU7 137660547 EC50 = 1500 nM T71230 CY89PF 137660705 IC50 > 1000 nM T71230 CH90KD 137660938 EC50 = 2 nM T71230 CF4DM3 137661087 EC50 = 19 nM T71230 CEO6T8 137661147 EC50 = 310 nM T71230 CVX3W8 137662168 IC50 = 0.094 nM T71230 CL4T0P 145964836 EC50 = 4000 nM T71230 CI73CT 145965177 EC50 = 320 nM T71230 CV7QC8 145965480 EC50 = 220 nM T71230 C8TWI9 145965832 EC50 = 380 nM T71230 C4H6ME 145966527 EC50 = 71 nM T71230 CP0M9O 145966606 EC50 = 1500 nM T71230 C1Y9ZM 145966623 EC50 = 340 nM T71230 CIP2M6 145969386 EC50 = 41 nM T71230 CHV5G4 145969643 EC50 = 720 nM T71230 CO5L6Q 145970751 EC50 = 320 nM T71230 C64ZOJ 145972874 EC50 = 850 nM T71230 CH7D0I 145972983 EC50 = 4000 nM T71230 CEJ7W1 145973560 EC50 = 900 nM T71230 C8U0QE 145973936 EC50 = 98 nM T71230 C89CMJ 145974446 EC50 = 620 nM T71230 CDT4Q8 145975421 EC50 = 110 nM T71230 CE58HG 145975579 EC50 = 420 nM T71230 C4Z9CJ 145976372 EC50 = 200 nM T71230 CQZM51 145977117 EC50 = 470 nM T71230 CJS6L4 145977163 EC50 = 0.1 nM T71230 CEK4I5 145977195 EC50 = 330 nM T71230 CH60XG 145978290 EC50 = 1000 nM T71230 CO3Q6I 145978338 EC50 = 780 nM T71230 COK19M 145978827 EC50 = 78 nM T71230 D0U3YQ 4551 IC50 = 36 nM T32821 CQ1A9K 384525 IC50 > 40000 nM T32821 CFET56 876233 IC50 = 1500 nM T32821 C3Z0DB 1361444 IC50 = 2500 nM T32821 CC68RW 2995979 IC50 = 2500 nM T32821 CF28EU 9799855 IC50 = 6 nM T32821 CG2Y6J 9880417 IC50 = 50 nM T32821 CLS4M1 9886720 IC50 = 60 nM T32821 CF6YE0 9901027 IC50 = 500 nM T32821 CRF1X2 9922214 IC50 = 1500 nM T32821 C8OX2Q 9924670 IC50 = 40 nM T32821 CSM8J6 9945339 IC50 = 12000 nM T32821 CUH89Z 9947061 IC50 = 15 nM T32821 CLBJ64 9967612 IC50 = 300 nM T32821 C2QX1C 9967803 IC50 = 160 nM T32821 CF2P1U 10022582 IC50 = 140 nM T32821 CMEN16 10110036 IC50 = 140 nM T32821 CM2F6C 10131537 IC50 = 11000 nM T32821 CM30PW 10154645 IC50 = 27 nM T32821 CFL24N 10200693 IC50 = 140 nM T32821 CV21QP 10201651 IC50 = 15 nM T32821 C3Z4RH 10267851 IC50 = 1000 nM T32821 C0SQI5 10269940 IC50 = 35 nM T32821 CND03G 10269987 IC50 = 170 nM T32821 CZN24R 10269990 IC50 = 45 nM T32821 C6NB3K 10271507 IC50 = 200 nM T32821 CY35XQ 10291040 IC50 = 190 nM T32821 CBGE57 10292766 IC50 = 60 nM T32821 C9DUN1 10406874 IC50 = 75 nM T32821 CT4E0S 11164727 IC50 = 17 nM T32821 CI96FD 11176626 IC50 = 10 nM T32821 CQ7WF8 11209986 IC50 = 240 nM T32821 CD9Y8U 11222131 IC50 = 6500 nM T32821 CA20CG 11245550 IC50 = 80 nM T32821 C1WD9Y 11257777 IC50 = 34 nM T32821 C7DNP9 11268641 IC50 = 50 nM T32821 CYHK07 11326288 IC50 = 50 nM T32821 CBMZ92 11337163 IC50 = 490 nM T32821 C29HAN 11348781 IC50 = 260 nM T32821 CF76JT 11350266 IC50 = 28 nM T32821 CLW6T5 11359913 IC50 = 22 nM T32821 C8J6HP 11360384 IC50 = 18000 nM T32821 CXEI65 11361007 IC50 = 24 nM T32821 C80RCA 11383098 IC50 = 99 nM T32821 CJDL86 11395628 IC50 = 8000 nM T32821 C0F7AD 11396375 IC50 = 18 nM T32821 C2F9BU 11405713 IC50 = 40 nM T32821 C2YOL0 11406630 IC50 = 31 nM T32821 CN68AO 11439833 IC50 = 54 nM T32821 CUP40B 11451948 IC50 = 28 nM T32821 CU5RP7 11461922 IC50 = 35000 nM T32821 COT4J0 11462697 IC50 = 20 nM T32821 CO4JC8 11462733 IC50 = 2100 nM T32821 C3P5VC 11475035 IC50 = 230 nM T32821 C3R2QG 11484569 IC50 = 29000 nM T32821 C9PWJ8 11485216 IC50 = 2050 nM T32821 CBJ0F9 11748922 IC50 = 800 nM T32821 CTVY73 12629814 IC50 = 1100 nM T32821 CQ3I7H 42606638 IC50 = 34 nM T32821 CZ4X7E 42606754 IC50 = 91 nM T32821 C68KSD 42606758 IC50 = 88 nM T32821 C1RH2W 42606875 IC50 = 750 nM T32821 CJ0I5Y 44282133 IC50 = 75 nM T32821 CGPE62 44282134 IC50 = 75 nM T32821 CM7GE5 44282210 IC50 = 550 nM T32821 C9KG0F 44282211 IC50 > 5000 nM T32821 C5DMP1 44282241 IC50 = 650 nM T32821 C7V1JZ 44282244 IC50 = 120 nM T32821 CH8D6L 44282273 IC50 = 5200 nM T32821 C7OMG1 44282334 IC50 > 64000 nM T32821 CG35SQ 44282339 IC50 = 9000 nM T32821 CIRE74 44282346 IC50 > 20000 nM T32821 CN1MQ2 44282363 IC50 = 70 nM T32821 C7WOS8 44282364 IC50 = 50 nM T32821 CM29RG 44282375 IC50 = 950 nM T32821 C8G1RF 44282398 IC50 = 100 nM T32821 CPI75A 44282399 IC50 > 20000 nM T32821 CCU50B 44282490 IC50 > 5000 nM T32821 CM9RI5 44282491 IC50 = 600 nM T32821 CJ2GA9 44282514 IC50 = 40000 nM T32821 C37BZC 44282538 IC50 > 5000 nM T32821 CT70FU 44282545 IC50 = 100 nM T32821 CYI86L 44282546 IC50 = 2000 nM T32821 CBC1U6 44282563 IC50 = 16000 nM T32821 CU9ZW4 44282564 IC50 = 12000 nM T32821 CBX17S 44282577 IC50 = 1400 nM T32821 CP4VN6 44282598 IC50 = 300 nM T32821 C45MDB 44282607 IC50 = 1500 nM T32821 C2I3ZP 44282613 IC50 = 15 nM T32821 CYS98J 44282662 IC50 > 20000 nM T32821 C0N6VM 44282711 IC50 = 500 nM T32821 CNQ38M 44282712 IC50 = 500 nM T32821 C7XL6Y 44282713 IC50 > 5000 nM T32821 C5QAI9 44282761 IC50 = 100 nM T32821 CGA4Y9 44282807 IC50 = 100 nM T32821 C74HAF 44282837 IC50 > 64000 nM T32821 CF3HT9 44282838 IC50 > 64000 nM T32821 CG8Z6R 44282854 IC50 = 64000 nM T32821 CJ40LB 44282932 IC50 = 64000 nM T32821 CYA8T2 44282941 IC50 = 800 nM T32821 C8E7SO 44282949 IC50 = 400 nM T32821 CQDB41 44282959 IC50 = 31000 nM T32821 CULY38 44282960 IC50 > 20000 nM T32821 C1R2VL 44282989 IC50 > 20000 nM T32821 CM8YI1 44313608 IC50 = 2300 nM T32821 CA4DW1 44313627 IC50 = 150 nM T32821 CX9TJ2 44313704 IC50 = 7000 nM T32821 C74TFB 44313707 IC50 = 640 nM T32821 CZ9WH4 44313708 IC50 = 970 nM T32821 CAL39F 44313822 IC50 = 2700 nM T32821 CQ59FH 44313823 IC50 = 16 nM T32821 C1CP6O 44313843 IC50 = 8300 nM T32821 C13UFJ 44313851 IC50 = 610 nM T32821 C71EQU 44313903 IC50 = 210 nM T32821 CXCZ82 44313942 IC50 = 17 nM T32821 CKJ39P 44313958 IC50 = 720 nM T32821 CBYE67 44313974 IC50 > 5000 nM T32821 CC23ZO 44313975 IC50 = 400 nM T32821 C0ODS2 44314040 IC50 = 120 nM T32821 C14ZLM 44314083 IC50 = 580 nM T32821 CO45SN 44314131 IC50 = 4900 nM T32821 C9SFB7 135436655 IC50 = 450 nM T32821 C2DY0I 136053632 IC50 = 10000 nM T22839 D0V3YT 10324367 IC50 > 10000 nM T22839 D0X9CH 3010818 IC50 = 30 nM T22839 CKJ1B7 382514 IC50 = 2720 nM T22839 CQ84MG 9917430 Ki = 1000000 nM T22839 C4L6CO 10093198 Ki = 290 nM T22839 CM50SP 11742283 IC50 = 1250 nM T22839 CQ8I1H 44353324 Ki = 660 nM T22839 C1RG9O 44353326 Ki = 160 nM T22839 C0D4CK 44353344 Ki = 1 nM T22839 C38RJF 44353357 Ki = 200 nM T22839 CQU69T 44353358 Ki = 14 nM T22839 CQH2K6 44353359 Ki > 1000000 nM T22839 C14NKU 44353376 Ki > 1500000 nM T22839 C3ZMS6 44353451 Ki = 850 nM T22839 CJW47S 44353453 Ki = 300 nM T22839 CD34OI 44353465 Ki = 0.58 nM T22839 C8XGW0 44353478 Ki = 4300 nM T22839 C7FHG9 44353531 Ki = 44 nM T22839 CB6GM1 44584127 IC50 = 1100 nM T22839 C4YAJ7 46228924 IC50 > 10000 nM T22839 CV0SF5 90664925 IC50 > 10000 nM T22839 D06FNK 122623 IC50 = 51.6 nM T22839 D06RRT 44353385 Ki = 41000 nM T22839 D0E9EH 44353386 Ki = 250 nM T36075 D03GOI 16134956 EC50 = 0.0657 nM T36075 D0H8WF 44278361 EC50 = 0.0439 nM T36075 D0V7SO 60151939 Ki = 3160 nM T36075 CZC24A 1259939 IC50 = 1288.25 nM T36075 CV0Q3D 1302369 IC50 = 602.56 nM T36075 C5HJV1 1401143 IC50 = 7200 nM T36075 C0GE2X 1619763 IC50 = 5754.4 nM T36075 C21HKV 1941609 IC50 = 691.83 nM T36075 CY4L6T 4143022 EC50 = 4100 nM T36075 CDUW70 9862981 EC50 = 2600 nM T36075 C31SPZ 9908249 EC50 = 5100 nM T36075 COV96E 9909122 EC50 = 1000 nM T36075 CGEJ24 9985625 IC50 > 10000 nM T36075 C6L7UO 10032265 IC50 = 17045 nM T36075 CR6NW9 10054055 IC50 = 4600 nM T36075 C62RYU 10144925 IC50 = 9323 nM T36075 CFD96W 10145290 IC50 = 21767 nM T36075 C08BCM 10257357 IC50 = 4900 nM T36075 CO2CQ7 11331120 IC50 = 4700 nM T36075 CC5WD2 11444850 IC50 = 5800 nM T36075 CJ4K2U 11456187 IC50 = 6700 nM T36075 CB59HM 11570626 IC50 > 10000 nM T36075 CE0CZ6 11764614 IC50 = 4879 nM T36075 CSZQ52 11764615 IC50 = 7731 nM T36075 CA8P2T 16007289 IC50 = 32 nM T36075 COF34S 16100296 IC50 = 1000 nM T36075 C53GHR 16100334 IC50 = 10773 nM T36075 CMV8T7 16135519 EC50 = 0.025 nM T36075 CS7PJ3 16139491 EC50 = 0.093 nM T36075 C5Y4XR 16141062 EC50 = 2.4 nM T36075 C8FN1X 16186241 EC50 = 846.8 nM T36075 C3IL9B 16199250 EC50 = 3.21 nM T36075 CV6TN8 16208189 EC50 = 22 nM T36075 CB8P6V 16209124 EC50 = 0.0009 nM T36075 C4GN5Q 20821266 IC50 = 3100 nM T36075 C2YH8O 20821269 EC50 = 4900 nM T36075 CO6YM4 20821273 EC50 = 7100 nM T36075 CF4DW8 22341045 EC50 = 175 nM T36075 CSLT25 22341047 EC50 = 214 nM T36075 CD0LN4 22341065 EC50 = 661 nM T36075 CQ1JI6 22341081 EC50 = 4300 nM T36075 CZ2NB3 22341083 EC50 = 2200 nM T36075 CZ8NE4 22341084 EC50 = 433 nM T36075 C0ASU1 22341109 EC50 = 2200 nM T36075 C0N2DQ 22341111 EC50 = 1800 nM T36075 CLZ4O1 22341128 EC50 = 1500 nM T36075 C2DFB4 22341129 EC50 = 1400 nM T36075 C2A3YE 22341131 EC50 = 1200 nM T36075 CP8WQ6 22341135 EC50 = 1200 nM T36075 CBM7I3 22341144 IC50 = 109 nM T36075 CQ7ST5 22341167 EC50 = 14000 nM T36075 CN9B4G 22341178 EC50 = 2600 nM T36075 CO67GH 22341180 EC50 = 3000 nM T36075 C1NYQ7 22341203 EC50 = 6300 nM T36075 C0SG1M 22341205 EC50 = 30000 nM T36075 C93KSJ 22341206 EC50 = 5000 nM T36075 C50RCH 23688809 IC50 = 21000 nM T36075 CLF63K 44290344 EC50 = 0.687 nM T36075 C7RSX3 44290345 EC50 = 0.0273 nM T36075 C5OLS1 44290396 EC50 = 0.022 nM T36075 C63VYZ 44290397 EC50 = 0.213 nM T36075 CC8DI0 44290523 EC50 = 0.0352 nM T36075 C92EPN 44290524 EC50 = 1.26 nM T36075 CPB8Q5 44290525 EC50 = 0.121 nM T36075 CN09YA 44290545 EC50 = 0.0301 nM T36075 C1EGK6 44290547 EC50 = 7 nM T36075 C6W9ZS 44290548 EC50 = 0.053 nM T36075 CW32MD 44290564 EC50 = 0.0363 nM T36075 C09HFM 44290565 EC50 = 0.0364 nM T36075 CA2Q8L 44290649 EC50 = 0.328 nM T36075 C2UAN7 44290650 EC50 = 0.054 nM T36075 C0F6IC 44290760 EC50 = 0.00789 nM T36075 CYI13E 44290761 EC50 = 0.21 nM T36075 CA5N2R 44290793 EC50 = 2.36 nM T36075 CF8OR9 44290794 EC50 = 0.41 nM T36075 C5ZC3B 44290820 EC50 = 0.0056 nM T36075 C5QOC9 44290821 EC50 = 0.116 nM T36075 CMOV30 44290898 EC50 = 0.194 nM T36075 CC3S4E 44290899 EC50 = 0.008 nM T36075 CEP3A8 44290900 EC50 = 3.05 nM T36075 CEX3V0 44290901 EC50 = 16.7 nM T36075 CF9CO8 44290915 EC50 = 0.115 nM T36075 C46RLN 44290916 EC50 = 0.00419 nM T36075 C53BVA 44290919 EC50 = 0.072 nM T36075 CSH4R9 44290924 EC50 = 0.113 nM T36075 CQ23OV 44290925 EC50 = 0.0844 nM T36075 C1PZ4N 44290999 EC50 = 0.154 nM T36075 C2BKE8 44291000 EC50 = 0.177 nM T36075 CRKV70 44291044 EC50 = 0.169 nM T36075 CKV3T8 44291066 EC50 = 0.135 nM T36075 C4J5IP 44291067 EC50 = 0.0272 nM T36075 C1CW0P 44394004 EC50 > 1000 nM T36075 C4E9KO 44394005 EC50 = 49 nM T36075 CEQW91 44394053 EC50 > 1000 nM T36075 C2M1HO 44394054 EC50 = 28 nM T36075 C2YT0B 44394055 EC50 = 37 nM T36075 C4YR2X 44394056 EC50 = 72 nM T36075 C2A1UO 44418950 IC50 = 100000 nM T36075 C80PUO 44442072 EC50 = 3300 nM T36075 CIH2N5 44442078 IC50 > 10000 nM T36075 CGT95I 44442081 IC50 > 10000 nM T36075 C40KZM 44442117 EC50 = 14000 nM T36075 CPU39C 44442131 EC50 = 5000 nM T36075 C8L1KQ 44442140 EC50 = 2200 nM T36075 C0E3QM 44449632 EC50 = 1400 nM T36075 CZ09MF 44587796 EC50 = 0.0056 nM T36075 C7KDL6 44598666 EC50 > 10000 nM T36075 C5OPK9 45381049 IC50 > 10000 nM T36075 CN0PU9 45381051 IC50 > 10000 nM T36075 CS5XO8 45381153 IC50 > 10000 nM T36075 C0RIG3 45381379 IC50 > 10000 nM T36075 C8UY2B 45381380 IC50 > 10000 nM T36075 CH13AF 45381381 IC50 > 10000 nM T36075 C5NQO0 45485567 EC50 = 545 nM T36075 CE4CY7 45485568 EC50 > 10000 nM T36075 CH90BO 45485569 EC50 = 787 nM T36075 C19HFB 45485570 EC50 = 480 nM T36075 C5UB8D 45485571 EC50 = 215 nM T36075 C5Q4YN 45485572 EC50 = 390 nM T36075 C16MHA 45485573 EC50 = 270 nM T36075 CR20VW 45485574 EC50 = 430 nM T36075 C9HA7K 45485575 EC50 = 148 nM T36075 CRWT51 45485576 EC50 = 87 nM T36075 C0VGH1 45485577 EC50 = 95 nM T36075 C70OKY 45485578 EC50 = 27 nM T36075 C8XEK5 45485579 EC50 = 93 nM T36075 C94GYF 45485580 EC50 = 35 nM T36075 CRF68L 45485581 EC50 = 965 nM T36075 CT18CM 45485582 EC50 = 7 nM T36075 CED20R 45485584 EC50 = 0.28 nM T36075 CQS1U6 45485585 EC50 = 0.087 nM T36075 CD48CL 49864564 EC50 = 0.015 nM T36075 C37MEV 49864565 EC50 = 0.026 nM T36075 CE9NY7 49864573 EC50 = 0.028 nM T36075 CWKH42 49864580 EC50 = 0.014 nM T36075 C1SG5P 49864615 EC50 = 0.013 nM T36075 CS3Y7O 51031037 IC50 > 10000 nM T36075 CRT2V5 53466721 IC50 > 10000 nM T36075 CO3KV0 53466723 IC50 > 10000 nM T36075 CZ9MH8 53469056 IC50 > 10000 nM T36075 CS0P9Y 53469058 IC50 > 10000 nM T36075 CN3O7H 53469258 IC50 > 10000 nM T36075 CD2X1W 53469443 IC50 > 10000 nM T36075 CU4R6T 53469628 IC50 = 2000 nM T36075 CU09OX 53469820 IC50 > 10000 nM T36075 CL7O5U 53469821 IC50 > 10000 nM T36075 C6TEK8 54765284 IC50 = 2600 nM T36075 C0T3KY 54765285 IC50 > 10000 nM T36075 C97STZ 56602804 IC50 > 10000 nM T36075 C1NG8L 56945626 EC50 = 202.5 nM T36075 CH8P3M 57391489 IC50 = 2300 nM T36075 CZ07MU 57391686 Ki = 816 nM T36075 CW4FM5 57393425 Ki = 9080 nM T36075 C7T0OK 57393426 Ki = 3340 nM T36075 CIU91X 57396928 Ki = 16500 nM T36075 C4AJ1G 57403703 IC50 = 2300 nM T36075 C81UIB 58352762 IC50 > 10000 nM T36075 CLW17X 58352803 IC50 > 10000 nM T36075 CTBN85 58352821 IC50 > 10000 nM T36075 CX83MS 58352834 IC50 > 10000 nM T36075 CFC36Q 58352858 IC50 > 10000 nM T36075 CXF21H 58352863 IC50 = 7800 nM T36075 C2I6KW 58352868 IC50 = 7300 nM T36075 CYXQ05 58352925 IC50 > 10000 nM T36075 CG4ZO9 58352935 IC50 > 10000 nM T36075 C9M3WT 58352937 IC50 > 10000 nM T36075 C2FN1G 58352938 IC50 > 10000 nM T36075 CW1UI5 58352940 IC50 = 6300 nM T36075 CG3RK7 58352952 IC50 = 4400 nM T36075 C12TUG 58352954 IC50 = 800 nM T36075 CH8MG0 58353013 IC50 = 6400 nM T36075 C94ITK 58353025 IC50 > 10000 nM T36075 C5PBI4 58353046 IC50 > 10000 nM T36075 C3GQ6I 58353063 IC50 = 5600 nM T36075 C9XR2K 58353067 IC50 > 10000 nM T36075 CBH52R 58353104 IC50 > 10000 nM T36075 CJ9F3R 58353126 IC50 > 10000 nM T36075 C5IXS0 58353156 IC50 = 3900 nM T36075 COCJ18 58353206 IC50 > 10000 nM T36075 CX95LQ 58353323 IC50 > 10000 nM T36075 C3KRI7 58353338 IC50 > 10000 nM T36075 C1YPO0 58353350 IC50 > 10000 nM T36075 C0SL8G 58353369 IC50 > 10000 nM T36075 CB9L4I 58353544 IC50 = 3100 nM T36075 CD57RC 58353625 IC50 > 10000 nM T36075 CMLO57 58353662 IC50 = 4300 nM T36075 CA7SI2 58353679 IC50 = 2200 nM T36075 C1IND2 58353695 IC50 > 10000 nM T36075 CLEZ12 58353778 IC50 > 10000 nM T36075 CG39KD 58353838 IC50 > 10000 nM T36075 CO0ZG7 58353839 IC50 > 10000 nM T36075 C4M1KY 58987474 EC50 = 0.12 nM T36075 C7KLY0 59337493 EC50 = 59 nM T36075 CPLU74 60170970 IC50 = 8200 nM T36075 CA0EO3 60171059 IC50 = 3300 nM T36075 CX5FQ8 68243839 IC50 > 10000 nM T36075 C3YW1K 68860750 IC50 > 1000 nM T36075 CX7S0D 70683012 EC50 > 1000 nM T36075 CIV6E4 70900317 IC50 > 10000 nM T36075 CT9DV6 71202679 IC50 = 140 nM T36075 C85ZLB 71202712 IC50 > 10000 nM T36075 CCY0M6 71202713 IC50 > 10000 nM T36075 CM4R1O 71202743 IC50 > 10000 nM T36075 C90NQH 71203427 IC50 > 10000 nM T36075 CF5WP9 71243005 IC50 > 10000 nM T36075 C6DQ1U 71243036 IC50 > 10000 nM T36075 C1K5TQ 71243097 IC50 > 10000 nM T36075 C3WCK2 73345594 EC50 = 24 nM T36075 C46KXM 73345595 EC50 = 15 nM T36075 C7MWC2 76314010 EC50 = 0.0049 nM T36075 C5TNY4 76314011 EC50 = 0.0261 nM T36075 CG7W9B 76314012 EC50 = 0.0015 nM T36075 CP02KO 76314013 EC50 = 0.003 nM T36075 CG23IQ 76317553 EC50 = 0.0336 nM T36075 CMS2X8 76317554 EC50 = 0.0368 nM T36075 CM84GO 76317555 EC50 = 0.0073 nM T36075 C01ARN 76317556 EC50 = 0.0181 nM T36075 CV2D0W 76321286 EC50 = 0.0032 nM T36075 CPWS73 76324900 EC50 = 0.0064 nM T36075 CIG21V 76324901 EC50 = 0.0032 nM T36075 C2L0UX 76324902 EC50 = 0.0065 nM T36075 CV8UI3 76328461 EC50 = 0.0038 nM T36075 C8IV6H 76328462 EC50 = 0.0219 nM T36075 CB4LI0 76332142 EC50 = 0.0034 nM T36075 CQ0AF2 76332143 EC50 = 0.0242 nM T36075 C1WTZ8 90655064 IC50 > 10000 nM T36075 C9U1WM 90655065 IC50 > 10000 nM T36075 CR26KU 90655066 IC50 > 10000 nM T36075 C1ON5Z 90655067 IC50 > 10000 nM T36075 CM6VG1 92239323 EC50 = 2041.74 nM T36075 CY2UI5 101891769 EC50 = 1300 nM T36075 C30HMF 118723386 EC50 = 6500 nM T36075 CQ1SC2 118723387 EC50 = 12022.64 nM T36075 CK9I4L 118723388 EC50 = 10232.93 nM T36075 CZHW75 118723389 EC50 = 14100 nM T36075 CW7XF9 118737073 Ki = 59 nM T36075 C9S1CB 118737074 EC50 = 10 nM T36075 CO8QT3 118737075 EC50 = 95 nM T36075 C10AWE 118737076 EC50 = 320 nM T36075 CTEH59 118737077 Ki = 320 nM T36075 C1D5XK 118737078 EC50 = 670 nM T36075 CEMW91 118737122 EC50 = 600 nM T36075 C1QD5W 118737123 EC50 = 190 nM T36075 C16CAT 118737124 EC50 = 81 nM T36075 CDB8N3 118737125 EC50 = 730 nM T36075 C0CKN7 118737126 EC50 = 110 nM T36075 CL7V5F 118737127 EC50 = 1.8 nM T36075 CI1PW5 118737128 EC50 = 0.73 nM T36075 C5Q1SJ 118737129 EC50 = 390 nM T36075 CA01TH 118737130 EC50 = 200 nM T36075 C94JKP 118737131 EC50 = 0.045 nM T36075 C7TDK6 122189729 EC50 = 0.0076 nM T36075 C63TKM 122189730 EC50 = 0.0171 nM T36075 CGN7X5 122189731 EC50 = 0.0037 nM T36075 CVT69Z 122189732 EC50 = 0.0709 nM T36075 CW1PB4 122189733 EC50 = 0.238 nM T36075 C3O5NW 122189734 EC50 = 0.0038 nM T36075 CPJ15R 122189735 EC50 = 0.0027 nM T36075 CI7M4S 122189736 EC50 = 0.0062 nM T36075 CP28FH 122189755 EC50 = 0.0192 nM T36075 CG8E7V 122189756 EC50 = 0.0111 nM T36075 C0U3LW 122189757 EC50 = 0.0147 nM T36075 CA3ZT7 122189758 EC50 = 0.0043 nM T36075 CL7JY5 122189759 EC50 = 0.0032 nM T36075 CV58LO 122189760 EC50 = 0.0048 nM T36075 C2S7EL 122189761 EC50 = 0.0426 nM T36075 CJ2V3L 122189762 EC50 = 0.0157 nM T36075 CE92RU 122189763 EC50 = 0.166 nM T36075 CST96G 122189764 EC50 = 0.0086 nM T36075 C93YLD 122189765 EC50 = 0.269 nM T36075 C1V7LD 122189766 EC50 = 0.0099 nM T36075 C46AYX 122189767 EC50 = 0.0048 nM T36075 CI94YP 122189768 EC50 = 0.0071 nM T36075 C24LBC 122189769 EC50 = 0.0056 nM T36075 CMQL59 122189770 EC50 = 0.0277 nM T36075 CELO20 122189771 EC50 = 0.0473 nM T36075 CNW52C 122189772 EC50 = 0.0278 nM T36075 CE15OZ 122189773 EC50 = 0.067 nM T36075 CD1BG4 122189774 EC50 = 0.0703 nM T36075 CT2L5M 122189775 EC50 = 0.0212 nM T36075 CV9M2K 122189776 EC50 = 0.0107 nM T36075 C5W4UB 122189777 EC50 = 5.99 nM T36075 C6AR3G 122189778 EC50 = 0.0115 nM T36075 CHZ56P 122189779 EC50 = 0.0244 nM T36075 C4KH1Y 122189780 EC50 = 0.007 nM T36075 CW68CO 122189781 EC50 = 0.0046 nM T36075 CKET80 122189782 EC50 = 0.0099 nM T36075 CN58PG 122189783 EC50 = 0.0409 nM T36075 C4H0NK 122189784 EC50 = 0.0027 nM T36075 CMC46Y 122189785 EC50 = 0.0418 nM T36075 C62PUR 122189786 EC50 = 0.159 nM T36075 CP0K2D 122189787 EC50 = 0.0873 nM T36075 C21SQE 122189788 EC50 = 0.0132 nM T36075 CDM8W4 122189789 EC50 = 0.0015 nM T36075 CV27CH 122189790 EC50 = 0.0675 nM T36075 CN3K6P 122189791 EC50 = 0.026 nM T36075 C78DEK 122195583 EC50 = 0.14 nM T36075 C61SKI 122195584 EC50 = 0.85 nM T36075 C5E0BI 122195585 EC50 = 430 nM T36075 CSI7U1 122195586 EC50 = 1400 nM T36075 C4Q6UM 122195587 EC50 = 13 nM T36075 CM5X8C 122195588 EC50 = 1 nM T36075 CKU95S 122195589 EC50 = 1000 nM T36075 CUM34W 122195590 EC50 = 2000 nM T36075 C3NP9U 122195591 EC50 = 390 nM T36075 CI81RE 122195592 EC50 = 19 nM T36075 CHOJ63 122195593 EC50 = 1000 nM T36075 CZV9R5 122195594 EC50 = 130 nM T36075 CU7JA0 122195595 EC50 = 2800 nM T36075 C3NZV9 122195596 EC50 = 2.4 nM T36075 C0ZN5Y 122195597 EC50 = 470 nM T36075 CQJP05 122195598 EC50 = 47 nM T36075 CYV3P9 122195599 EC50 = 360 nM T36075 C38TMY 122195600 EC50 = 2.5 nM T36075 C98TOP 122195601 EC50 = 2000 nM T36075 CP53LS 122195602 EC50 = 0.47 nM T36075 C7X4WI 122195805 EC50 = 430 nM T36075 CF38XW 122195806 EC50 = 5000 nM T36075 CC95FV 122195807 EC50 = 1600 nM T36075 CI10MH 122195808 EC50 = 16000 nM T36075 C89MRN 122195809 EC50 = 69 nM T36075 CG37UP 122195810 EC50 = 7500 nM T36075 C83WVN 122195811 EC50 = 850 nM T36075 C94TXK 122195812 EC50 = 1150 nM T36075 C01LJA 122195813 EC50 > 1000 nM T36075 C1XID0 127027153 EC50 = 0.0329 nM T36075 CS0X5Z 127028394 EC50 = 0.0636 nM T36075 C4A3XT 127029032 EC50 = 0.0766 nM T36075 CTH8D2 127048230 EC50 > 1000 nM T36075 C6IME2 127048235 EC50 = 60 nM T36075 CYQ06U 127048242 EC50 > 1000 nM T36075 CSJ4E0 127048563 EC50 > 1000 nM T36075 C06PAY 127048570 EC50 > 1000 nM T36075 CIC5N9 127048573 EC50 > 1000 nM T36075 C0QD6C 127048580 EC50 > 1000 nM T36075 COAX23 127048585 EC50 > 1000 nM T36075 C9AYL1 127048586 EC50 > 1000 nM T36075 CQJ4I9 127048907 EC50 = 100 nM T36075 CNFT67 127048913 EC50 = 16 nM T36075 C2T1RK 127048919 EC50 > 1000 nM T36075 CZM2P6 127048924 EC50 = 45 nM T36075 CU6B7T 127048925 EC50 = 8.9 nM T36075 C9CBY0 127049246 EC50 > 1000 nM T36075 C3EZ1Q 127049553 EC50 > 1000 nM T36075 CHF48Z 127049554 EC50 > 1000 nM T36075 CZ04YP 127049559 EC50 > 1000 nM T36075 CF8E4Y 127049561 EC50 > 1000 nM T36075 CTND43 127049562 EC50 > 1000 nM T36075 C2YK9U 127049569 EC50 = 80 nM T36075 CU0WT7 127049891 EC50 > 1000 nM T36075 C8O3ZH 127049892 EC50 > 1000 nM T36075 C91XKU 127049900 EC50 > 1000 nM T36075 C91XMF 127049904 EC50 > 1000 nM T36075 C05KIM 127049905 EC50 > 1000 nM T36075 CGZI28 127049907 EC50 = 83 nM T36075 CI3X9N 127050190 EC50 > 1000 nM T36075 CJ8MO0 127050192 EC50 > 1000 nM T36075 CLQE96 127050193 EC50 > 1000 nM T36075 C2T3NQ 127050489 EC50 > 1000 nM T36075 C52ROH 127050497 EC50 = 300 nM T36075 CUY7X9 127050499 EC50 > 1000 nM T36075 C6X9AW 127050816 EC50 > 1000 nM T36075 CJ79TN 127050817 EC50 > 1000 nM T36075 CQKE41 127050829 EC50 > 1000 nM T36075 C6VX5B 127051083 EC50 > 1000 nM T36075 CO0MQ4 127051084 EC50 = 39 nM T36075 CCVE81 127051086 EC50 = 180 nM T36075 C1URK5 127051088 EC50 > 1000 nM T36075 CG4D0F 127051089 EC50 > 1000 nM T36075 CQT03Z 127051091 EC50 = 90 nM T36075 C8AWI0 127051094 EC50 > 1000 nM T36075 COS48H 127051377 EC50 > 1000 nM T36075 CX8AU4 127051382 EC50 > 1000 nM T36075 C21PCY 127051386 EC50 > 1000 nM T36075 CYN56P 127051391 EC50 > 1000 nM T36075 C97SOU 127051393 EC50 > 1000 nM T36075 CG7W2D 127051708 EC50 = 40 nM T36075 CV96NH 127051710 EC50 > 1000 nM T36075 CQ7G8U 127051715 EC50 > 1000 nM T36075 CAJ0F5 127051716 EC50 > 1000 nM T36075 CZL51Q 127051717 EC50 > 1000 nM T36075 C2AWU3 127051718 EC50 > 1000 nM T36075 CK41ZJ 127052018 EC50 > 1000 nM T36075 CS0HY2 127052019 EC50 = 56 nM T36075 CE63MT 127052022 EC50 > 1000 nM T36075 CC7DM5 127052029 EC50 = 32 nM T36075 C4PO0G 127052034 EC50 > 1000 nM T36075 C5CUZ1 127052341 EC50 > 1000 nM T36075 C9QC7T 127052344 EC50 > 1000 nM T36075 C95WZR 127052351 EC50 = 70 nM T36075 CKQG87 127052643 EC50 > 1000 nM T36075 CAO0W7 127052645 EC50 > 1000 nM T36075 CN0LF8 127052647 EC50 > 1000 nM T36075 C0I1LV 127052648 EC50 > 1000 nM T36075 CW4V7K 127052654 EC50 = 130 nM T36075 C5K3JR 127052936 EC50 > 1000 nM T36075 CXJ7C0 127052938 EC50 > 1000 nM T36075 C3RTO1 127052943 EC50 = 120 nM T36075 C75QMW 127052944 EC50 = 110 nM T36075 CY9L1H 127052945 EC50 > 1000 nM T36075 COB7C9 127052953 EC50 > 1000 nM T36075 C2BR6S 134611040 EC50 = 12 nM T36075 C3ZEH8 137319706 EC50 = 600 nM T36075 CP3B6J 137632640 Ki > 50 nM T36075 C1NDQ2 137633001 EC50 = 0.004 nM T36075 CX5MS9 137633159 EC50 = 0.0052 nM T36075 C6PC5L 137633723 EC50 = 0.011 nM T36075 C5PC4U 137633868 EC50 = 0.023 nM T36075 C3JFZ5 137634115 EC50 = 0.0174 nM T36075 C3YHG5 137634214 EC50 = 0.0172 nM T36075 CY40VR 137634741 EC50 = 0.0254 nM T36075 CVU64X 137634800 EC50 = 0.021 nM T36075 CDC1Y8 137635047 EC50 = 0.148 nM T36075 CO1BK4 137635623 EC50 = 0.035 nM T36075 C60LYD 137635778 Ki = 34 nM T36075 CB4I7O 137638423 EC50 = 0.0022 nM T36075 CMQU03 137639569 Ki = 10 nM T36075 CWVF96 137639902 Ki > 50 nM T36075 CYM17E 137640544 EC50 = 0.074 nM T36075 CQMX23 137640594 EC50 = 0.0558 nM T36075 CG3FR1 137640853 EC50 = 0.068 nM T36075 CIS76Q 137641519 Ki = 16 nM T36075 CEX6K4 137642925 EC50 = 0.0039 nM T36075 C72VWS 137643463 EC50 = 1.9 nM T36075 CQ7E1C 137643772 EC50 = 0.0153 nM T36075 CU70VG 137644146 EC50 = 0.02 nM T36075 CPNM90 137645271 EC50 = 0.006 nM T36075 CJX36T 137646811 EC50 = 300 nM T36075 CEG1J7 137647087 EC50 = 0.013 nM T36075 CBR2K3 137647238 EC50 = 0.118 nM T36075 CNIX49 137647741 EC50 = 0.05 nM T36075 C0CB6I 137648322 EC50 = 0.05 nM T36075 CLPM69 137648373 EC50 = 0.0313 nM T36075 CPJ26D 137649424 EC50 = 0.1 nM T36075 CK2JM7 137649897 EC50 = 0.0082 nM T36075 CI72XO 137650720 EC50 = 0.0007 nM T36075 C9EPK4 137651037 EC50 = 0.547 nM T36075 C0YHE3 137651113 Ki > 50 nM T36075 C3M7WP 137652582 Ki > 50 nM T36075 C8YN7M 137653668 EC50 = 0.054 nM T36075 CS8WM2 137654780 EC50 = 0.0058 nM T36075 CL6BC4 137655542 EC50 = 0.009 nM T36075 CT8R6B 137656322 EC50 = 0.0018 nM T36075 CC82TK 137656477 Ki > 50 nM T36075 C0L1DH 137656580 EC50 = 0.35 nM T36075 C1HWA8 137656776 EC50 = 0.522 nM T36075 C7EST1 137656784 EC50 = 20 nM T36075 C6I1UA 137658847 EC50 = 0.0012 nM T36075 C5ZD1M 137659233 EC50 = 0.0222 nM T36075 CYE08C 137660014 EC50 = 0.041 nM T36075 C4ZT1U 137660531 EC50 = 0.0222 nM T36075 C1CJM5 137661058 Ki > 50 nM T36075 C15YGR 137661214 EC50 = 0.221 nM T36075 CZK81P 137661599 EC50 = 0.0209 nM T36075 CEA4T0 137662138 EC50 = 0.041 nM T36075 CJ5FS6 137662302 EC50 = 1.63 nM T36075 CU1P4W 145948755 EC50 > 1000 nM T36075 CGY3Q0 145948765 EC50 > 1000 nM T36075 CAXE41 145948867 EC50 > 1000 nM T36075 CB3D9P 145948868 EC50 > 1000 nM T36075 CR2M7E 145948881 EC50 = 21 nM T36075 CIDG54 145948888 EC50 > 1000 nM T36075 CZ70FB 145948890 EC50 = 8.8 nM T36075 CHD30J 145948895 EC50 > 1 nM T36075 CJI6Y0 145948896 EC50 = 0.1886 nM T36075 C3GOA2 145948898 EC50 = 0.0237 nM T36075 CTV1K7 145948929 EC50 = 10 nM T36075 CMCH73 145948934 EC50 > 1 nM T36075 C7Z2XN 145948936 EC50 = 0.0053 nM T36075 C8AH3T 145948941 EC50 > 1 nM T36075 CBR0M6 145948943 EC50 = 0.0209 nM T36075 C2X9BL 145948944 EC50 = 0.0284 nM T36075 CQ6I0F 145948972 EC50 > 1000 nM T36075 C5QB1Z 145948975 EC50 > 1000 nM T36075 CES8B1 145948994 EC50 > 1 nM T36075 C3BNV8 145949006 EC50 > 1 nM T36075 CQ29TZ 145949291 EC50 = 0.86 nM T36075 C4LE9A 145949559 EC50 = 5.86 nM T36075 CB8O0I 145950198 EC50 = 8.96 nM T36075 C8K1TP 145950470 EC50 = 112.03 nM T36075 CIFH84 145951037 EC50 = 3.3 nM T36075 CG52YC 145952042 EC50 = 16.16 nM T36075 C7MC0S 145953388 EC50 = 6.14 nM T36075 CGLY87 145953555 EC50 = 3.58 nM T36075 C9A1LQ 145953718 EC50 = 4.54 nM T36075 C7CK8M 145953834 EC50 = 1.84 nM T36075 C3A6GO 145956482 EC50 = 1.72 nM T36075 C6OFU3 145956601 EC50 = 88.23 nM T36075 CW5PY0 145956908 EC50 = 10.31 nM T36075 C0M6PJ 145957642 EC50 = 29.4 nM T36075 CLKX02 145958107 EC50 = 31.93 nM T36075 C96YSZ 145958355 EC50 = 0.94 nM T36075 CSQ0B2 145958772 EC50 = 1.4 nM T36075 CGNW71 145959528 EC50 = 3 nM T36075 CW1X9P 145959606 EC50 = 51.72 nM T36075 C7HZY1 145959966 EC50 = 1.6 nM T36075 C7N3KL 145960401 EC50 = 0.0053 nM T36075 C92BLJ 145960433 EC50 = 0.0025 nM T36075 C0X5MI 145960850 EC50 = 0.0018 nM T36075 CT1JB9 145961416 EC50 = 3.01 nM T36075 C1ZNU5 145961751 EC50 = 0.0048 nM T36075 CW90YV 145962263 EC50 = 0.0525 nM T36075 CN9CR1 145962270 EC50 = 0.0022 nM T36075 CA29XQ 145962515 EC50 = 0.0064 nM T36075 CVQ62L 145962554 EC50 = 0.0022 nM T36075 C97HKT 145962593 EC50 = 0.0039 nM T36075 CGO8V1 145962872 EC50 = 0.0014 nM T36075 C0ADY2 145962907 EC50 = 0.008 nM T36075 CLO0S4 145967618 EC50 = 0.03 nM T36075 C05PHX 145967716 EC50 = 0.0056 nM T36075 CQDI82 145967926 EC50 = 0.09 nM T36075 C3JW1P 145968295 EC50 = 0.039 nM T36075 C0T1ZE 145968501 EC50 = 0.068 nM T36075 C0ZTW8 145968513 EC50 = 0.093 nM T36075 C8GIF3 145968867 EC50 = 0.0198 nM T36075 CMB10N 145969232 EC50 = 0.003 nM T36075 C5J8HP 145969289 EC50 = 0.02 nM T36075 CUOK61 145969452 EC50 = 0.0263 nM T36075 C7UZT9 145969722 EC50 = 0.015 nM T36075 CS36QG 145969945 EC50 = 0.022 nM T36075 C3AI9B 145970440 EC50 = 0.14 nM T36075 CX0C6A 145970613 EC50 = 0.04 nM T36075 CI2H8F 145970697 EC50 = 0.0093 nM T36075 CCZ9K7 145970869 EC50 = 0.004 nM T36075 CDB15L 145971098 EC50 = 0.115 nM T36075 CN4Z2C 145971132 EC50 = 0.002 nM T36075 CV4F0E 145974582 EC50 = 2 nM T36075 CN6U7X 145979055 EC50 = 16.3 nM T36075 CXLG95 145979356 EC50 = 9.6 nM T36075 CJ20ZC 145979450 EC50 = 6.2 nM T36075 CU0TG9 145979952 EC50 = 2.8 nM T36075 C28RZK 145981006 EC50 = 16.8 nM T36075 CW61LE 145983653 EC50 = 4.1 nM T36075 CV93OQ 145986807 EC50 = 0.0061 nM T36075 C12KQR 145986934 EC50 = 3.1 nM T36075 C9L1DZ 145987268 EC50 = 0.0143 nM T36075 CC3Y2Z 145987495 EC50 = 0.003 nM T36075 CI92LE 145988245 EC50 = 12.1 nM T36075 C6G8LE 145989624 EC50 = 11.8 nM T36075 CE1O2V 145989690 EC50 = 7.3 nM T36075 C8JM2S 145989854 EC50 = 5.2 nM T36075 C2EBS6 145990393 EC50 = 23.5 nM T36075 CMT69Z 145990732 EC50 = 6.9 nM T36075 CHB90P 145992609 EC50 = 5.4 nM T36075 CDS5V3 155516067 EC50 = 5 nM T36075 CO1B9Q 155517307 EC50 = 3.981 nM T36075 C0L3MD 155525234 EC50 = 1.5 nM T36075 CH5JY2 155526075 EC50 = 0.0202 nM T36075 C5MJI7 155532030 EC50 = 0.0182 nM T36075 C02WEF 155535132 EC50 = 1.585 nM T36075 CN85FI 155541367 EC50 = 1.2 nM T36075 CKI6O4 155543961 EC50 = 0.0064 nM T36075 CB52ZK 155547392 EC50 = 1 nM T36075 C1XVJ3 155547905 EC50 = 0.07 nM T36075 CPG12J 155550533 EC50 = 0.0169 nM T36075 CS8BW0 155560523 EC50 = 0.17 nM T36075 CG94TV 155567378 EC50 = 0.021 nM T36075 C08ZCY 155567532 EC50 = 5 nM T17758 D05HXX 5526 Ki = 2000000 nM T17758 D05PHH 3447 IC50 = 431 nM T17758 D0AZ8C 5213 IC50 = 21000 nM T17758 D0FT4R 107706 IC50 > 2000 nM T17758 D0I0RJ 16231 IC50 = 2400 nM T17758 D0K8KX 5280343 IC50 = 12100 nM T17758 D00EPS 449051 Ki = 20 nM T17758 D00LOB 9866964 Ki > 26000 nM T17758 D01MUU 183797 Ki = 6300 nM T17758 D03KGH 9830667 Ki = 410 nM T17758 D0G0YZ 9885167 Ki = 37 nM T17758 D02INZ 2387 Ki = 2330 nM T17758 D03QJN 9895762 Ki > 17000 nM T17758 D08INO 9895194 Ki = 960 nM T17758 D0K1PR 1747 Ki = 79.43 nM T17758 D0W9PG 124704 IC50 > 1000000 nM T17758 C71WRJ 1503 Ki = 3600 nM T17758 CY5B9C 1504 Ki = 400 nM T17758 C2KE5Q 1508 Ki = 2400 nM T17758 C9TMQ4 1725 IC50 = 7000 nM T17758 C4S1PB 4300 Ki = 6000 nM T17758 CL1T7V 4301 Ki = 2700 nM T17758 CUSM50 11974 Ki = 1570 nM T17758 CTJ0C5 13624 IC50 = 200000 nM T17758 C0YU1V 16157 IC50 = 20000 nM T17758 C5P3TH 65130 Ki = 14400 nM T17758 CQ0MW7 68540 Ki = 7000 nM T17758 C8CQW2 73742 Ki = 50118.72 nM T17758 CLHY62 76630 IC50 > 1000000 nM T17758 CT28FD 80002 Ki = 20600 nM T17758 C1UNL9 90295 Ki = 50118.72 nM T17758 CK9AZ0 122670 Ki = 131000 nM T17758 C6MQD0 124952 IC50 = 26000 nM T17758 CRMX39 159363 IC50 > 1000000 nM T17758 C50XVJ 159772 Ki = 744731.97 nM T17758 C1BHS3 193409 Ki = 5900 nM T17758 CO97IC 194530 IC50 > 1000000 nM T17758 CZP0Y1 204101 Ki > 13000 nM T17758 CIR92Q 409363 Ki = 258821.29 nM T17758 C32CWP 409364 Ki = 15595.53 nM T17758 CZ1QL5 411406 Ki = 1980 nM T17758 CB9VP7 432298 Ki = 1950 nM T17758 CR4KE5 445844 Ki = 9 nM T17758 CU6X2A 445847 Ki = 190 nM T17758 C5UX1L 447478 Ki = 190 nM T17758 CVND42 447482 Ki = 250 nM T17758 C4OKV5 447486 Ki = 550 nM T17758 CC9G5O 447490 Ki = 11 nM T17758 CR2DX3 447496 Ki = 250 nM T17758 COYS31 447502 Ki = 2800 nM T17758 CVI28M 447508 Ki = 55 nM T17758 CS09BE 447510 Ki = 280 nM T17758 C87GLP 447540 Ki = 32 nM T17758 C87OTC 447733 Ki = 39.81 nM T17758 CF6D4B 447734 Ki = 25.12 nM T17758 CHT05K 447735 Ki = 48 nM T17758 CFMI91 448548 Ki = 36 nM T17758 C5QKC3 448605 Ki = 0.62 nM T17758 CX5MS1 448610 Ki = 30 nM T17758 CO01KD 456168 Ki = 17800 nM T17758 C0P9RD 459983 Ki = 4470 nM T17758 C3NB2K 459984 Ki = 8000 nM T17758 C2ZBC5 583065 Ki = 50118.72 nM T17758 COK61H 639391 IC50 = 484 nM T17758 C53FNM 674593 IC50 = 120 nM T17758 C45NBS 674629 IC50 = 1500 nM T17758 C21HDC 674632 IC50 = 170 nM T17758 CG2UK8 674633 IC50 = 18400 nM T17758 CX1W4S 674635 IC50 = 28300 nM T17758 C9PI4L 674639 IC50 = 4700 nM T17758 CI9LH0 674642 IC50 = 32300 nM T17758 CBX3U0 674652 IC50 = 2500 nM T17758 COD8V2 674657 IC50 = 2500 nM T17758 CW5ZA1 680939 IC50 = 1100 nM T17758 C8BQU5 833517 IC50 = 33600 nM T17758 CLR3H1 899247 IC50 = 24900 nM T17758 CBRI54 1036823 IC50 = 41100 nM T17758 C49RWG 1549311 Ki = 38904.51 nM T17758 C4ZUJ5 2757788 Ki = 6067.36 nM T17758 C7W8YC 3010979 Ki = 380 nM T17758 C76VAR 3010993 Ki = 125.89 nM T17758 CSO6N0 3010999 Ki = 63.1 nM T17758 CTO48W 3081948 IC50 = 5000 nM T17758 C85WXS 3085183 IC50 = 2000 nM T17758 C1DU3P 3580940 Ki = 54300 nM T17758 CIR7L6 3621644 Ki = 676000 nM T17758 C5PJK7 3631189 Ki = 90700 nM T17758 C9HEB1 3675673 IC50 = 50000 nM T17758 CJDR03 3963048 IC50 = 2500 nM T17758 C4DT8I 4475489 Ki = 9300 nM T17758 CCS5F4 4475490 Ki = 48000 nM T17758 CB9WS0 4653788 Ki = 56000 nM T17758 CV8W5G 4713320 Ki = 19000 nM T17758 CRK73Q 4713323 Ki = 73000 nM T17758 CQC05H 4713327 Ki = 19000 nM T17758 CJC7N6 4713329 Ki = 41000 nM T17758 CY5KR6 4713353 Ki = 58000 nM T17758 CHS9T0 4713355 Ki = 16000 nM T17758 C9A0IZ 4713356 Ki = 38000 nM T17758 CVT61D 4713357 Ki = 2000 nM T17758 C3HQK8 4713365 Ki = 26000 nM T17758 CD02VO 4713366 Ki = 1300 nM T17758 C2G7OB 4713372 Ki = 12000 nM T17758 C2I4MP 4713404 Ki = 56000 nM T17758 C81KBP 4713415 Ki = 17000 nM T17758 C3Z7HR 4713420 Ki = 800000 nM T17758 CHF96N 5173985 Ki = 418793.57 nM T17758 C8I0VG 5289529 Ki = 630 nM T17758 CQ26VM 5289531 Ki = 640 nM T17758 C7SYK9 6102731 IC50 = 5900 nM T17758 CN2B6S 6852211 Ki = 1100 nM T17758 C4OP6M 7038665 IC50 > 62000 nM T17758 CX34ZD 9549214 Ki > 1800 nM T17758 C39JGW 9797957 IC50 = 320 nM T17758 C6JDM9 9799627 Ki = 6.3 nM T17758 CM7Q0R 9799840 Ki = 280 nM T17758 CU05FV 9800468 Ki = 350 nM T17758 CYN72M 9800469 Ki = 1100 nM T17758 C7E8KD 9800470 Ki = 700 nM T17758 CI6U9Z 9802199 Ki = 44000 nM T17758 CKA6C4 9802514 Ki = 8 nM T17758 CY5F7E 9803095 Ki = 1180 nM T17758 C1FIN6 9804775 IC50 > 130 nM T17758 C2AXV0 9809479 Ki > 13000 nM T17758 CF9S0B 9815838 Ki = 8700 nM T17758 CLW6S3 9816370 Ki = 2900 nM T17758 CKN89B 9822176 Ki = 115000 nM T17758 C1D4EC 9822928 Ki = 5.8 nM T17758 CPB20R 9826345 Ki = 430 nM T17758 CGN48U 9827867 IC50 = 60000 nM T17758 CM05AF 9838290 Ki = 125.89 nM T17758 C2I1QV 9843613 Ki = 440 nM T17758 C8Z5TX 9843775 Ki = 9.9 nM T17758 C5H4DR 9846031 Ki = 430 nM T17758 CS9HQ0 9850467 IC50 = 335 nM T17758 CPOT59 9867086 Ki = 280 nM T17758 CL6QS0 9868922 Ki = 7.7 nM T17758 CDU85Y 9871868 Ki = 4500 nM T17758 C45CVJ 9881397 Ki = 600 nM T17758 C2F5NS 9884570 Ki = 20 nM T17758 CQP0V2 9886960 Ki = 80 nM T17758 C5B4VE 9890102 Ki = 180 nM T17758 CKDP84 9895193 Ki = 410 nM T17758 CQ5H2C 9903519 Ki = 1000 nM T17758 C73DNO 9908936 Ki = 287000 nM T17758 CMC95R 9910164 Ki = 508 nM T17758 CD5LQ0 9910982 Ki > 200000 nM T17758 C13XPD 9912856 Ki = 16 nM T17758 CC0D5H 9915041 Ki > 13000 nM T17758 CFO1K9 9922130 Ki = 21000 nM T17758 CLZ53G 9922131 Ki = 12000 nM T17758 C8C6UI 9929077 Ki = 102 nM T17758 C2UX6D 9930716 Ki = 7.4 nM T17758 CG3B1P 9935390 Ki = 280 nM T17758 CNE25D 9935474 Ki = 1.4 nM T17758 CL2NV0 9935925 IC50 > 870 nM T17758 CC9QH7 9937406 IC50 = 600 nM T17758 C8F5CW 9937921 Ki > 19000 nM T17758 C8LR4T 9938917 Ki > 13000 nM T17758 CDT95S 9939426 Ki = 650 nM T17758 C1K5WI 9948854 Ki = 170 nM T17758 CFK05S 9949275 Ki = 100 nM T17758 C1RHT8 9949886 Ki = 38 nM T17758 CTWX05 9950966 Ki = 240 nM T17758 CEI68D 9951603 Ki = 280 nM T17758 CYP6S7 9952109 Ki = 10 nM T17758 C4F3NM 9952313 Ki = 310 nM T17758 CPR2L8 9952552 Ki = 280 nM T17758 C4CX9Q 9953631 Ki = 1500 nM T17758 CW7TZ6 9953704 IC50 = 23.1 nM T17758 CX85LD 9954980 Ki > 14000 nM T17758 CCQE85 9956843 Ki = 1.6 nM T17758 CYLI95 9956922 Ki = 2.6 nM T17758 CKIP10 9987251 IC50 = 4.3 nM T17758 C2PQV5 10021506 Ki = 44000 nM T17758 CX4TI5 10029172 Ki = 390 nM T17758 CFCT67 10053115 Ki = 400 nM T17758 CZH3W7 10094378 Ki > 200000 nM T17758 CQP65H 10095093 Ki > 1000000 nM T17758 C17CDJ 10096845 IC50 = 3.1 nM T17758 CK1W7N 10110404 Ki = 610 nM T17758 CW4RZ5 10116936 IC50 > 450 nM T17758 C5E0SY 10126451 Ki = 125.89 nM T17758 C5VJE7 10131165 Ki = 4830 nM T17758 CR03NV 10131788 Ki = 41000 nM T17758 CS2G4T 10140847 Ki = 18 nM T17758 C31QAL 10143532 Ki > 13000 nM T17758 C7L5IJ 10157296 Ki = 91 nM T17758 CL7U8P 10181581 Ki = 28 nM T17758 C7PC2K 10185292 IC50 > 170 nM T17758 CFIH78 10185526 IC50 = 15500 nM T17758 CEP79T 10216518 Ki = 50 nM T17758 CC2EA1 10219529 Ki = 32300 nM T17758 C8V1AY 10225952 Ki = 40 nM T17758 CG3C0S 10243600 Ki = 120 nM T17758 C2XHG8 10248900 Ki = 91000 nM T17758 CUX40O 10258264 Ki = 410 nM T17758 C32CBS 10262708 Ki = 3130 nM T17758 CSX60M 10264543 Ki = 350 nM T17758 C0J1TD 10278414 Ki = 2 nM T17758 CNAX45 10287785 Ki = 142 nM T17758 CZM97W 10293977 Ki = 23000 nM T17758 C5EDW1 10294146 Ki = 100 nM T17758 CA9NP3 10305055 Ki = 50.12 nM T17758 C1LCO8 10335742 Ki = 138 nM T17758 C9XUD8 10347489 IC50 = 1210 nM T17758 CJ0O5P 10367277 IC50 = 6999 nM T17758 CNJ03F 10374840 Ki = 61659.5 nM T17758 CSC52L 10390341 Ki = 31000 nM T17758 CJNV62 10391699 IC50 > 33000 nM T17758 C84THX 10424840 Ki = 103 nM T17758 CJTH60 10432907 Ki = 22 nM T17758 C6AZ8B 10435038 Ki > 1000000 nM T17758 CWG91R 10472893 Ki = 86000 nM T17758 CFS2U9 10474680 Ki = 3400 nM T17758 CQ8C1S 10480047 Ki = 60 nM T17758 CEI65Z 10483775 Ki = 2100 nM T17758 CFP53Y 10502109 IC50 > 33000 nM T17758 CU8N3V 10578280 IC50 > 10000 nM T17758 C8SUZ9 10624948 Ki > 1000000 nM T17758 CEJ14F 10624997 Ki = 34000 nM T17758 CR5EX8 10648196 Ki = 15000 nM T17758 CPWH69 10648370 Ki = 110000 nM T17758 CW1G9B 10672666 IC50 > 10000 nM T17758 C5VB1U 10695159 Ki > 1000000 nM T17758 CGYR23 10696955 Ki = 32000 nM T17758 CGP79W 10697355 IC50 = 5300 nM T17758 CPGV87 10718240 Ki > 1000000 nM T17758 CL7RC5 10742017 IC50 > 33000 nM T17758 CKOQ35 10767421 Ki > 1000000 nM T17758 C3IN8W 10815545 Ki = 140000 nM T17758 CVQE76 10816339 Ki = 28000 nM T17758 CLB15C 10871563 Ki = 100 nM T17758 CW7Q2U 10895700 IC50 > 250000 nM T17758 CQTC02 10903566 Ki = 550 nM T17758 C8OA1L 10946869 Ki = 13000 nM T17758 C2TBO9 10959252 Ki = 360 nM T17758 C43SNO 11004109 Ki = 100 nM T17758 CC39SB 11009950 Ki = 55000 nM T17758 CYZL25 11015002 Ki = 43 nM T17758 CD9WJ8 11057540 Ki = 55 nM T17758 C2Y6VW 11057779 Ki = 25 nM T17758 C3HNB2 11068806 Ki = 280 nM T17758 CAD15G 11149953 Ki = 1900 nM T17758 C8DVG9 11152403 Ki = 5020 nM T17758 CJ4X7R 11158066 IC50 = 61 nM T17758 C6LVG4 11186243 Ki = 38 nM T17758 CTX9F3 11188793 Ki = 123 nM T17758 CR0SZ8 11218419 Ki = 8700 nM T17758 C50NYT 11222761 Ki = 517 nM T17758 CGC9O1 11227852 IC50 = 1100 nM T17758 CLA93S 11237163 Ki > 14000 nM T17758 C4MJX6 11243198 Ki = 7980 nM T17758 CHLK70 11244460 Ki = 326 nM T17758 CHAN28 11245701 Ki = 167 nM T17758 CEP9B5 11254287 IC50 > 62000 nM T17758 CPB32N 11257364 Ki = 104 nM T17758 CX9Z7A 11277660 IC50 = 17000 nM T17758 CB1GW5 11285134 IC50 = 4100 nM T17758 CGP3B1 11290529 Ki = 82 nM T17758 C86DZB 11292119 Ki = 23.5 nM T17758 CK6RO7 11312725 Ki = 15500 nM T17758 C91GMZ 11317532 Ki > 100000 nM T17758 C34GUA 11326599 Ki = 100 nM T17758 C6CDN3 11347670 Ki = 736 nM T17758 CLY5G8 11350400 Ki = 35.5 nM T17758 CR8NW9 11351302 Ki > 14000 nM T17758 C6JXY9 11361521 Ki = 161 nM T17758 CTJ1Z2 11361949 Ki = 26.5 nM T17758 CNX6W1 11399761 IC50 = 1600 nM T17758 CGW75B 11419694 Ki = 86 nM T17758 CIQH43 11445130 IC50 = 532 nM T17758 C9O4NF 11450922 Ki = 139 nM T17758 C63LIR 11473486 Ki = 63 nM T17758 CVI82D 11479420 Ki = 16000 nM T17758 CJZ09N 11512593 Ki = 19000 nM T17758 C28BMR 11513105 Ki = 3600 nM T17758 CRNU10 11534959 Ki = 4600 nM T17758 CD1A6T 11542037 Ki = 260 nM T17758 CA8KD7 11542038 Ki = 810 nM T17758 CBP69L 11557024 Ki = 1700 nM T17758 CCG84F 11563457 Ki = 10500 nM T17758 CV46NL 11563632 Ki = 25000 nM T17758 CEAZ46 11569930 Ki = 2100 nM T17758 C3TJ7M 11570580 Ki = 1900 nM T17758 C6RHD8 11570700 Ki = 1800 nM T17758 C1DN2L 11570759 Ki = 56000 nM T17758 C6FG8V 11577055 Ki = 2300 nM T17758 CIY34V 11577968 Ki = 18000 nM T17758 CJ38EP 11577970 Ki = 8900 nM T17758 C7MF9N 11578158 Ki = 320 nM T17758 CTSK74 11584729 Ki = 3600 nM T17758 C1RQ6P 11592130 Ki = 8000 nM T17758 CBC84M 11592593 Ki = 1100 nM T17758 C7ZS8L 11592600 Ki = 6100 nM T17758 C7QTY8 11606981 Ki = 1200 nM T17758 CU07NO 11607091 Ki = 1200 nM T17758 CL9TZ2 11614477 Ki = 620 nM T17758 CB4O2Q 11621579 Ki = 12000 nM T17758 CD3R1E 11627899 Ki = 11000 nM T17758 CB9P0Q 11628768 Ki = 600 nM T17758 CO3Q9N 11635973 Ki = 1500 nM T17758 CRX98P 11636026 Ki = 26000 nM T17758 CW10CL 11642802 Ki = 1300 nM T17758 C2W5XF 11656797 Ki = 820 nM T17758 C4SAR0 11657278 Ki = 31000 nM T17758 CVQ16C 11664107 Ki = 2100 nM T17758 CPZG49 11664334 Ki = 43000 nM T17758 CT9E0G 11664643 Ki = 820 nM T17758 CWV87X 11671266 Ki = 1500 nM T17758 CE0A6N 11671776 Ki = 1200 nM T17758 C85GCY 11671956 Ki = 2500 nM T17758 C1DHO6 11678360 Ki = 2200 nM T17758 C4IBO3 11678764 Ki = 3400 nM T17758 C69YSR 11693028 Ki = 1200 nM T17758 CCQY30 11693049 Ki = 7700 nM T17758 CPFW75 11699600 Ki = 2300 nM T17758 C3VS2H 11699903 Ki = 3600 nM T17758 CNV09Z 11699913 Ki = 2300 nM T17758 CKQ4O2 11721188 Ki = 6900 nM T17758 C4UB2X 11721375 Ki = 4000 nM T17758 C70AGR 11738687 Ki = 233 nM T17758 CQ5U8H 11739438 Ki = 15.85 nM T17758 C05TNR 11754398 Ki = 47000 nM T17758 C8GJO7 11754872 IC50 > 33000 nM T17758 C6ZT1D 11763794 IC50 = 250 nM T17758 C7JLR1 11774107 Ki = 28 nM T17758 CQ0T5X 11779259 IC50 = 2000 nM T17758 CR2E9T 11782463 Ki = 35 nM T17758 CNO67W 11798089 Ki > 1000000 nM T17758 C98ZOR 11824040 Ki = 3200 nM T17758 CYX74A 11824584 Ki = 490 nM T17758 CN6RP0 11983358 IC50 = 455 nM T17758 CZ15UV 12253678 Ki = 103000 nM T17758 C4FH3L 12253733 Ki = 292000 nM T17758 C7GO9F 12319196 IC50 > 1000000 nM T17758 C3OHB0 12336481 Ki = 136000 nM T17758 CX9Q2G 12420538 Ki = 30690.22 nM T17758 CBDW65 12459438 Ki = 12000 nM T17758 C8SG1D 13041565 Ki = 29000 nM T17758 CQ8OU1 13755335 IC50 > 10000 nM T17758 C7FUH3 14045773 IC50 > 1000000 nM T17758 CV7UY6 14298047 IC50 > 1000000 nM T17758 C94BTA 14346967 Ki = 1448771.85 nM T17758 CYW90B 15230351 IC50 = 500 nM T17758 C19ARJ 15984063 Ki > 150000 nM T17758 CLP2D3 16004672 Ki > 5000 nM T17758 CA8Y1K 16046152 Ki > 13000 nM T17758 CNBJ60 16046153 Ki > 13000 nM T17758 C5TBL6 16049247 IC50 = 3.1 nM T17758 C9BH4X 16086308 IC50 = 2.6 nM T17758 CF1V2N 16086310 IC50 = 5 nM T17758 C9JX7U 16086312 IC50 = 1.5 nM T17758 CK7IM0 16086316 IC50 = 6.2 nM T17758 CT9QM5 16086318 IC50 = 4.4 nM T17758 CXO65R 16086320 IC50 = 6 nM T17758 C3EUJ6 16086336 IC50 = 4 nM T17758 CR9EN3 16086338 IC50 = 5.8 nM T17758 CR7B3D 16086340 IC50 = 6.9 nM T17758 C90CXM 16086342 IC50 = 5.8 nM T17758 C7T5AI 16086344 IC50 = 6.6 nM T17758 CJZ63N 16086346 IC50 = 7 nM T17758 C05XAN 16086348 IC50 = 5 nM T17758 CACN42 16086349 IC50 = 6.7 nM T17758 CN6CJ2 16220264 IC50 = 8670 nM T17758 CZB89F 16657876 Ki = 19 nM T17758 CS9W6K 16657879 Ki = 66 nM T17758 C09DTL 16657882 Ki = 22 nM T17758 C3WX9G 16657950 Ki = 27 nM T17758 CBPA54 16658031 Ki = 7.4 nM T17758 C7JHS4 16658108 Ki = 11 nM T17758 CCVQ54 16658112 Ki = 330 nM T17758 C6V7DS 16658181 Ki = 111 nM T17758 C0TW3X 16658183 Ki = 23 nM T17758 CDA03H 16658245 Ki = 160 nM T17758 CG5RL7 16658246 Ki = 54 nM T17758 C1I6KE 16658248 Ki = 11 nM T17758 CPNJ21 16658250 Ki = 14 nM T17758 CLRQ75 16658288 Ki = 67 nM T17758 C5Q6JS 16658289 Ki = 30 nM T17758 CG98OH 16658290 Ki = 10 nM T17758 CO3ZV4 16658354 Ki = 130 nM T17758 CSMU45 16658355 Ki = 550 nM T17758 C46CDF 16658356 Ki = 59 nM T17758 C8DI4G 16658357 Ki = 58 nM T17758 C0Y4ZW 16658407 Ki = 29 nM T17758 C6NR2O 16658408 Ki = 31 nM T17758 CB6PC9 16658409 Ki = 21 nM T17758 CBX83S 16658633 Ki = 71 nM T17758 C8TP6S 16658679 Ki = 330 nM T17758 CZ58FK 16658680 Ki = 48 nM T17758 C0ZKU2 16658740 Ki = 43 nM T17758 C70XKG 16658742 Ki = 54 nM T17758 CQDT69 16658745 Ki = 35 nM T17758 C48TLQ 16658805 Ki = 28 nM T17758 CU60AH 16718671 IC50 = 7.2 nM T17758 COAB94 16718712 IC50 = 8 nM T17758 CU28CE 16718713 IC50 = 3.4 nM T17758 CA41KL 16718715 IC50 = 1600 nM T17758 CLI4D7 16718757 IC50 = 3.5 nM T17758 C2SFC0 16718759 IC50 = 67 nM T17758 CC20PS 16718760 IC50 = 6.6 nM T17758 CCKO80 16718762 IC50 = 26.5 nM T17758 CTZ74D 16718807 IC50 = 114 nM T17758 C37MRI 16718808 IC50 = 7 nM T17758 CW2LR9 18536775 Ki = 89000 nM T17758 CO9X8T 18536789 Ki = 70 nM T17758 CAI56P 18536809 Ki = 3900 nM T17758 CLD01Q 18536856 Ki = 160 nM T17758 CIM3R5 18536877 Ki = 277000 nM T17758 C3FPX2 18536880 Ki = 94000 nM T17758 C3GZT0 18536889 Ki = 90 nM T17758 C89CGD 18536897 Ki = 170 nM T17758 CZL15E 18536922 Ki = 270000 nM T17758 CZON79 18536933 Ki = 5490 nM T17758 CBF3V5 18536936 Ki = 531 nM T17758 CC5B4E 18536939 Ki = 910 nM T17758 C4BE0N 18536965 Ki > 28000 nM T17758 CH95RX 18536993 Ki = 1460 nM T17758 C1I6MF 18537001 Ki = 94000 nM T17758 CR0MI2 18537006 Ki = 164000 nM T17758 CJ2DQ9 18537029 Ki = 546000 nM T17758 C4E5PK 18537035 Ki = 2500 nM T17758 C6CDS5 18537037 Ki = 327000 nM T17758 C3OAT2 18537046 Ki = 180 nM T17758 CE38OR 18537047 Ki = 154000 nM T17758 CMW92K 18537075 Ki = 1110 nM T17758 C1CZ3E 18537077 Ki = 200 nM T17758 C64WAO 18537081 Ki = 982000 nM T17758 CSKV81 18537116 Ki = 80 nM T17758 CE9UY2 18537117 Ki = 120000 nM T17758 CB5GF8 18537172 Ki = 400 nM T17758 CUL10T 18537184 Ki = 1740000 nM T17758 CCN9K2 18537190 Ki = 108000 nM T17758 CRJ81N 18537194 Ki = 470000 nM T17758 C2P7AX 18537198 Ki = 130000 nM T17758 C0MZ5R 18537208 Ki = 110 nM T17758 C2A9JS 18537241 Ki = 442000 nM T17758 C58RBI 18537258 Ki = 305000 nM T17758 CP3J4F 18537281 Ki = 1420 nM T17758 CT6S1B 18537287 Ki = 161000 nM T17758 CI1AJ2 18537289 Ki = 58 nM T17758 CT9D4Y 18537290 Ki = 641000 nM T17758 CE64GP 18537293 Ki = 110 nM T17758 C6PR7W 18537298 Ki = 138000 nM T17758 CI9S7G 18537305 Ki = 640 nM T17758 C9O6AC 18537308 Ki = 200 nM T17758 CZ5WN1 18537312 Ki > 34000 nM T17758 CBY7U6 18537322 Ki = 2500 nM T17758 CZO7I0 18537342 Ki = 178000 nM T17758 CVHS18 18537399 Ki = 180 nM T17758 CES05C 18537429 Ki = 1620 nM T17758 CBL1Z8 18537461 Ki = 660 nM T17758 CJH4D2 18537468 Ki = 152000 nM T17758 CF9C8R 18537480 Ki = 1400 nM T17758 CYO70H 18545754 Ki = 196000 nM T17758 C6ML3J 18680125 Ki = 293 nM T17758 CX36SV 18771291 Ki = 300 nM T17758 C24CAY 18771297 Ki = 1920 nM T17758 CK71LJ 19841587 Ki = 6486.34 nM T17758 CBD5Y9 20229530 Ki = 26500 nM T17758 CE07DR 20690188 Ki = 370 nM T17758 CZ6KH9 20760195 Ki > 13000 nM T17758 CRGN82 21186404 Ki = 794.33 nM T17758 CT4B3N 21192441 Ki = 83 nM T17758 C2I8WX 21192489 Ki = 9300 nM T17758 C2Z9NT 21192495 Ki = 200 nM T17758 CA07SQ 21434854 Ki = 388000 nM T17758 C5UB8M 21705171 Ki = 209000 nM T17758 CMHT69 21706803 Ki = 630.96 nM T17758 CDG96S 21706810 Ki = 2300 nM T17758 C2KW0G 21706820 Ki = 125.89 nM T17758 CS4PZ6 21706825 Ki = 1995.26 nM T17758 CZQ1L4 21706843 Ki = 630.96 nM T17758 CJX8A1 21706877 Ki = 398.11 nM T17758 C2CGS8 21706927 Ki = 251.19 nM T17758 CF4EN3 21706931 Ki = 6309.57 nM T17758 C6DOH8 21706937 Ki = 3162.28 nM T17758 CU9C6N 21706939 Ki = 398.11 nM T17758 CA63IO 21706943 Ki = 530 nM T17758 C45SAH 21706953 Ki = 1995.26 nM T17758 C80JYP 21707001 Ki = 82000 nM T17758 CQTZ60 21707028 Ki = 630.96 nM T17758 C3H6XW 21707065 Ki = 1258.93 nM T17758 C61RMQ 21707067 Ki = 794.33 nM T17758 C5JD2U 21707080 Ki = 450 nM T17758 CIF9G4 21707110 Ki = 1584.89 nM T17758 C2OW6C 21707157 Ki = 251.19 nM T17758 C4RO3K 22018948 Ki = 100000 nM T17758 CNOT37 22098976 Ki = 1318256.74 nM T17758 C4YL7S 22556963 Ki = 270 nM T17758 C9VXC8 22556983 Ki = 1600 nM T17758 C1Q9XU 23278259 IC50 = 19000 nM T17758 CRX19I 23646295 Ki > 13000 nM T17758 CCRD27 23646312 Ki > 40000 nM T17758 C1WE6B 23646315 Ki > 13000 nM T17758 CSFH79 23646622 Ki = 150 nM T17758 C35HJA 23646623 Ki = 270 nM T17758 C7E4SA 23646732 Ki = 190 nM T17758 CU4RQ3 23653529 IC50 = 40000 nM T17758 CN2WM8 23653530 IC50 = 5200 nM T17758 CXV0K2 23653531 IC50 = 1300 nM T17758 C3RP7C 23653532 IC50 = 520 nM T17758 C06EVU 23653533 IC50 = 72 nM T17758 CKH4O5 24180463 Ki > 14000 nM T17758 C7AYO1 24748789 IC50 = 260 nM T17758 CVO5L6 24748791 IC50 = 900 nM T17758 CUAY58 24749175 IC50 = 4.2 nM T17758 CL2PU5 24750417 IC50 = 7.7 nM T17758 CU23HR 24774191 IC50 = 35000 nM T17758 CZ2P7E 24774192 IC50 = 1600 nM T17758 CWX10T 24774275 IC50 = 460 nM T17758 C8Q3KE 24774276 IC50 = 23000 nM T17758 C0N8LA 24774277 IC50 = 2700 nM T17758 CT6W3A 24774278 IC50 = 720 nM T17758 CN0ZW3 24999867 Ki > 1000 nM T17758 CEM32W 25001205 Ki > 1000 nM T17758 CAO2V4 25030840 Ki = 3300 nM T17758 CU82IO 25030929 Ki = 3700 nM T17758 C7MCT6 25031099 Ki = 880 nM T17758 C5PO7A 25031100 Ki = 17000 nM T17758 CH7Z1K 25031101 Ki = 2100 nM T17758 CEW9X2 25031102 Ki = 2500 nM T17758 C9NC4S 25031541 Ki = 2600 nM T17758 CK5R8Q 25032200 Ki = 3300 nM T17758 CG8HY2 25032202 Ki = 7400 nM T17758 CH76XK 25032204 Ki = 9200 nM T17758 CI8HE3 25138142 IC50 > 33000 nM T17758 CR5UN9 25141167 IC50 = 26 nM T17758 C2H4PJ 25166809 Ki > 28000 nM T17758 CG76TR 25181493 Ki = 10000 nM T17758 CWY5P1 28082833 IC50 > 62000 nM T17758 CS5J2O 28742032 Ki = 280000 nM T17758 C19OGX 44278104 Ki = 927 nM T17758 C1YMQ2 44278528 Ki = 272000 nM T17758 C2XA9D 44278529 Ki = 100000 nM T17758 CY9X2D 44278565 Ki = 145000 nM T17758 C0B1XM 44278581 Ki = 141000 nM T17758 C8Y9JZ 44284991 Ki > 63 nM T17758 CMZ71H 44284992 Ki = 23 nM T17758 C5NU9L 44285118 Ki = 540 nM T17758 CU9G2F 44285211 Ki = 15 nM T17758 C0FPN1 44285253 Ki = 33 nM T17758 C9N1ZL 44285281 Ki > 4.3 nM T17758 C5PX3O 44285312 Ki > 48 nM T17758 C9LRW8 44285352 Ki = 140 nM T17758 C3HR9X 44285724 Ki = 92000 nM T17758 C3QD4W 44287797 Ki > 200000 nM T17758 C5W7SA 44287798 Ki > 200000 nM T17758 C02ARM 44287937 Ki > 200000 nM T17758 CP90NM 44288029 Ki > 200000 nM T17758 CYA94B 44294210 Ki = 9960 nM T17758 C0O2PG 44295723 Ki = 350 nM T17758 C8AY9O 44296035 Ki = 8600 nM T17758 CQ51FN 44296074 Ki = 2300 nM T17758 C3DG0L 44296128 Ki = 320 nM T17758 CPF86Z 44296129 Ki = 2300 nM T17758 C38SDX 44296130 Ki = 12400 nM T17758 C1WU8B 44296135 Ki = 350 nM T17758 CPBH13 44297808 Ki = 40700 nM T17758 CFSN46 44297819 Ki = 83800 nM T17758 CXE86U 44297829 Ki = 5470 nM T17758 CF78HW 44297834 Ki = 147000 nM T17758 CMV68W 44297835 Ki = 53300 nM T17758 C6YUK2 44297837 Ki = 173000 nM T17758 CK01TP 44297841 Ki = 37700 nM T17758 CROG80 44297850 Ki = 10000 nM T17758 C9LGN2 44297867 Ki = 62000 nM T17758 CPM76K 44298377 Ki = 1500 nM T17758 CCYA19 44298389 Ki = 1280 nM T17758 CEX5K8 44298390 Ki = 2100 nM T17758 C8KJS9 44298438 Ki = 2000 nM T17758 C5V7HP 44298457 Ki = 16100 nM T17758 COA52Y 44298458 Ki = 90200 nM T17758 CQP29R 44298459 Ki = 9310 nM T17758 C4VT7F 44298473 Ki = 770 nM T17758 CQ9VT1 44298501 Ki = 16400 nM T17758 C76URK 44298504 Ki = 490 nM T17758 CJU7B0 44298507 Ki = 690 nM T17758 CS1I3Q 44298510 Ki = 1600 nM T17758 C2P7QZ 44298511 Ki = 2130 nM T17758 COU03N 44298523 Ki = 730 nM T17758 C13TMY 44298524 Ki = 550 nM T17758 CRS39A 44298525 Ki = 770 nM T17758 C84VKY 44298526 Ki = 166300 nM T17758 CV6Q8C 44298538 Ki = 920 nM T17758 C29MVU 44303719 Ki = 27000 nM T17758 C3FB4I 44303721 Ki > 75000 nM T17758 CQLA16 44303733 Ki = 24000 nM T17758 C5RZL0 44303743 Ki = 180 nM T17758 CTE75P 44303769 Ki = 650 nM T17758 C16GOI 44303778 Ki = 6000 nM T17758 C26ZUK 44303789 Ki = 3100 nM T17758 CN6V9A 44303803 Ki = 1000 nM T17758 C67ZRW 44303804 Ki = 8500 nM T17758 CB38WA 44303805 Ki = 190 nM T17758 CL0U1A 44303806 Ki = 1700 nM T17758 CVO2D9 44303808 Ki = 44000 nM T17758 C0JZY5 44303810 Ki = 8000 nM T17758 CFJ4W3 44303811 Ki = 2600 nM T17758 CE0R9A 44303824 Ki = 10000 nM T17758 C5YF7O 44303839 Ki = 13000 nM T17758 C2LY4T 44303843 Ki = 600 nM T17758 C3HXW6 44303858 Ki = 8 nM T17758 CYW9S8 44303912 Ki = 230 nM T17758 CIQZ37 44303925 Ki = 180 nM T17758 CJN72A 44303933 Ki = 450 nM T17758 CXCY31 44303935 Ki = 280 nM T17758 C4SN8T 44304006 Ki = 5500 nM T17758 CL16JC 44304046 Ki = 27000 nM T17758 CAM6R0 44304047 Ki = 20000 nM T17758 CR4V0L 44304084 Ki = 700 nM T17758 CG37DH 44304086 Ki = 220 nM T17758 C7UJH1 44304087 Ki = 85 nM T17758 CG0R8N 44304097 Ki = 250 nM T17758 CJ80KE 44304098 Ki = 4600 nM T17758 CG8TI6 44304099 Ki = 1600 nM T17758 C9W8QC 44304100 Ki = 8500 nM T17758 CE31BF 44304104 Ki = 300 nM T17758 C9XIO1 44304105 Ki > 75000 nM T17758 C83YIU 44304139 Ki = 8000 nM T17758 CP5S9K 44304192 Ki = 42000 nM T17758 CKD98A 44304353 Ki = 60000 nM T17758 CZEX59 44311229 IC50 = 970 nM T17758 CKP5W7 44311564 IC50 = 34 nM T17758 CM8N6K 44317510 IC50 = 8400 nM T17758 CN08YB 44331576 Ki = 36000 nM T17758 C98RIJ 44331596 Ki = 10600 nM T17758 CLZ0I6 44331643 Ki = 19000 nM T17758 C58VKT 44331672 Ki = 267000 nM T17758 CKB3M5 44331988 Ki > 100000 nM T17758 CV6R7F 44331989 Ki > 100000 nM T17758 CMI8V5 44332049 Ki = 40000 nM T17758 C7Y8IG 44334488 Ki = 2.1 nM T17758 CIE0O8 44334703 Ki = 4600 nM T17758 CHL01I 44334805 Ki = 8.5 nM T17758 CRT4G3 44335601 Ki = 49000 nM T17758 C7Z9WL 44335624 Ki = 58000 nM T17758 CHWY63 44336861 Ki = 3500 nM T17758 C0YO9D 44336901 Ki = 28000 nM T17758 C4SE8Q 44336925 Ki = 860 nM T17758 CYC7S4 44336980 Ki = 2500 nM T17758 CY45FN 44336995 Ki = 52000 nM T17758 C2V8OP 44336996 Ki = 33000 nM T17758 C0DIH9 44336997 Ki = 1300 nM T17758 C73QCK 44337001 Ki = 52000 nM T17758 C5OEX1 44337004 Ki = 7800 nM T17758 C2S4HW 44337018 Ki = 4400 nM T17758 C3W2DF 44337028 Ki = 5400 nM T17758 CR2C7L 44337052 Ki = 5100 nM T17758 C7A3ZN 44337099 Ki = 12000 nM T17758 CO7FI5 44337101 Ki = 19000 nM T17758 C18AZH 44337119 Ki = 4800 nM T17758 CND8F1 44339118 Ki = 310 nM T17758 CQ37SV 44339192 Ki > 100000 nM T17758 CCA37E 44339231 Ki = 830 nM T17758 C89EZV 44339232 Ki = 580 nM T17758 C8JQA9 44339233 Ki = 4930 nM T17758 CH6IY7 44339247 Ki = 3620 nM T17758 CU52DY 44339260 Ki = 640 nM T17758 CNQ2B0 44339261 Ki = 1000 nM T17758 C3XI4S 44339270 Ki = 400 nM T17758 CU20ZI 44339271 Ki = 340 nM T17758 C98MCJ 44339277 Ki = 800 nM T17758 CJ34AW 44339278 Ki = 660 nM T17758 C7PW4I 44339280 Ki = 1300 nM T17758 C7CAT2 44339282 Ki = 2340 nM T17758 C27PNV 44339304 Ki = 180 nM T17758 CQR82M 44339377 Ki = 1400 nM T17758 CD28KW 44339411 Ki = 82 nM T17758 CX3B5S 44339419 Ki = 9 nM T17758 CBU40W 44339439 Ki = 100 nM T17758 CU0PN1 44339441 Ki = 490 nM T17758 CXL2Q8 44341827 Ki = 494000 nM T17758 CX9MJ6 44356715 Ki = 10 nM T17758 CSJK97 44356716 Ki = 18730 nM T17758 C9REH6 44356739 Ki = 6000 nM T17758 CO8T4Z 44356858 Ki = 7830 nM T17758 CT4P3J 44363891 Ki = 169 nM T17758 CJAK97 44363903 Ki = 1520 nM T17758 C7IJY6 44367340 Ki = 1400 nM T17758 C7ZIU8 44367346 Ki = 35000 nM T17758 C5SD9G 44367355 Ki > 1000000 nM T17758 CHB97U 44367367 Ki = 25000 nM T17758 C8YP2H 44367372 Ki = 1600 nM T17758 CWD01E 44367382 Ki > 1000000 nM T17758 CX72JW 44367411 Ki = 34000 nM T17758 CTOC70 44367422 Ki = 40000 nM T17758 CXB28Z 44367430 Ki = 78000 nM T17758 CFY5B6 44367435 Ki = 49000 nM T17758 CYDQ04 44367444 Ki = 55000 nM T17758 C39FZP 44372663 Ki = 2200 nM T17758 C9I0BE 44372667 Ki = 500 nM T17758 CQLA75 44372683 Ki = 1500 nM T17758 CKFN05 44372724 Ki = 82000 nM T17758 CTD36H 44372738 Ki = 9000 nM T17758 CI6MQ5 44372778 Ki = 9200 nM T17758 CFH41R 44372839 Ki = 48 nM T17758 C9COY7 44372840 Ki = 61000 nM T17758 C34AWY 44372863 Ki = 4000 nM T17758 CZE15A 44372864 Ki = 1200 nM T17758 C7X5BE 44372865 Ki = 13 nM T17758 C1UEX9 44372875 Ki = 9600 nM T17758 C2E6TP 44372889 Ki = 490 nM T17758 C36XWM 44372903 Ki = 43 nM T17758 C3MX8T 44383176 Ki = 280 nM T17758 CN5WK2 44383197 Ki = 500 nM T17758 C26ZWY 44383362 Ki = 3060 nM T17758 CZB2T4 44383365 Ki = 480 nM T17758 C6RON5 44383439 Ki = 1840 nM T17758 CJZE25 44383520 Ki = 520 nM T17758 C0HNA8 44383819 Ki = 1020 nM T17758 C71AKQ 44383933 Ki = 6000 nM T17758 CE3QL1 44384306 Ki = 1600 nM T17758 COQH07 44385725 IC50 = 10.3 nM T17758 CX9W5Z 44385770 IC50 = 5.1 nM T17758 C7MXA5 44385833 IC50 = 19 nM T17758 C8F2RG 44386052 IC50 = 12.4 nM T17758 C5YF1O 44386205 IC50 = 101 nM T17758 C52MCK 44386366 IC50 = 11 nM T17758 CBG1U6 44386478 IC50 = 261 nM T17758 CWTU45 44386804 IC50 > 2500 nM T17758 CA0W2K 44386893 IC50 > 2500 nM T17758 CAY27D 44392382 Ki = 65 nM T17758 C9DNW6 44392384 Ki = 731 nM T17758 C2SQ1C 44392401 Ki = 281 nM T17758 C4VKE9 44392403 Ki = 10 nM T17758 CYL52J 44392413 Ki = 5 nM T17758 CN8CJ3 44392416 Ki = 622 nM T17758 CY0C3N 44392417 Ki = 1258.93 nM T17758 CE42KB 44392423 Ki = 47 nM T17758 CORK28 44392427 Ki = 263 nM T17758 C2J8BD 44392431 Ki = 548 nM T17758 CAF3G9 44392450 Ki = 198 nM T17758 C5CS1Z 44412395 IC50 = 370 nM T17758 C0P2OJ 44412397 IC50 = 2600 nM T17758 C6GNZ2 44412399 IC50 = 7800 nM T17758 CF8XV9 44412471 IC50 = 98 nM T17758 C5AME3 44412473 IC50 = 204 nM T17758 CSW2A9 44412496 IC50 = 53 nM T17758 C1MQ4U 44412499 IC50 = 208 nM T17758 C3BX5Y 44412781 Ki > 150000 nM T17758 CF5XO4 44413343 Ki = 1600 nM T17758 CTD42X 44413355 Ki = 6600 nM T17758 C9KQM2 44413356 Ki = 8200 nM T17758 CQDX92 44413619 Ki = 870 nM T17758 CPN1S0 44416248 IC50 = 8 nM T17758 C4A8IF 44422910 IC50 = 6910 nM T17758 COUZ56 44426215 Ki > 5000 nM T17758 C3F2PN 44426216 Ki > 5000 nM T17758 CZ91LH 44426217 Ki > 5000 nM T17758 CEV53U 44426218 Ki > 5000 nM T17758 C8O6HV 44426219 Ki = 150000 nM T17758 CJH6E4 44426220 Ki > 5000 nM T17758 C3E2FT 44426221 Ki > 5000 nM T17758 CW3G0D 44426222 Ki > 5000 nM T17758 CN6VL5 44426224 Ki > 5000 nM T17758 CG9XF0 44426226 Ki > 5000 nM T17758 CQ7CF9 44426227 Ki > 5000 nM T17758 CL4N6J 44426228 Ki > 5000 nM T17758 CJ3B7D 44426229 Ki > 5000 nM T17758 C5Q8HB 44426230 Ki > 5000 nM T17758 C6RNO7 44426232 Ki > 5000 nM T17758 CCGR09 44426234 Ki > 5000 nM T17758 CD06OJ 44426235 Ki > 5000 nM T17758 CR4D0U 44426236 Ki > 5000 nM T17758 CIT7D5 44426237 Ki > 5000 nM T17758 CW71LJ 44426238 Ki > 5000 nM T17758 CY5Z6P 44426239 Ki > 5000 nM T17758 CI0N7E 44426240 Ki > 5000 nM T17758 C35VBM 44426241 Ki > 5000 nM T17758 C0LIG6 44426243 Ki > 5000 nM T17758 C9V2JR 44426244 Ki > 5000 nM T17758 C72TBW 44426245 Ki > 5000 nM T17758 CZ2GS7 44426246 Ki > 5000 nM T17758 CPKM97 44426247 Ki > 5000 nM T17758 C1MVS4 44426248 Ki > 5000 nM T17758 C5W1RJ 44426249 Ki > 5000 nM T17758 C8H5OR 44426250 Ki > 5000 nM T17758 C8BE9L 44426251 Ki > 5000 nM T17758 CT6C5J 44426252 Ki > 5000 nM T17758 CCN6T9 44426253 Ki > 5000 nM T17758 C1UYG6 44426254 Ki > 5000 nM T17758 CVO5Q1 44432538 Ki > 14000 nM T17758 C2SMQ6 44433791 Ki = 34000 nM T17758 CR16BF 44434808 Ki > 14000 nM T17758 CQIX73 44434809 Ki > 14000 nM T17758 C5R8HJ 44434815 Ki > 14000 nM T17758 COG34X 44434818 Ki > 14000 nM T17758 C9T1DP 44434835 Ki > 14000 nM T17758 C30CFX 44436704 IC50 = 840 nM T17758 CEW6G1 44569299 Ki = 6600 nM T17758 C9JNT3 44569300 Ki = 8700 nM T17758 C9XE7Q 44569301 Ki > 1000000 nM T17758 CZI8D7 44569333 Ki > 1000000 nM T17758 CR4CP6 44569359 Ki = 129000 nM T17758 C9JF7W 44569667 Ki = 3800 nM T17758 C61IJB 44569732 Ki = 5200 nM T17758 CR36MB 44569733 Ki = 3000 nM T17758 CE25UL 44569767 Ki = 8100 nM T17758 C0CZ4I 44569768 Ki = 3200 nM T17758 CIR4M0 44569769 Ki = 8300 nM T17758 C02SHD 44569811 Ki = 12000 nM T17758 CG3LE9 44569812 Ki = 12000 nM T17758 CCU7V0 44569813 Ki = 11000 nM T17758 C8BR6E 44569843 Ki = 8600 nM T17758 C7Q9BH 44569844 Ki = 9600 nM T17758 CZ35OW 44569845 Ki = 14000 nM T17758 CHV9C1 44569846 Ki = 6900 nM T17758 C5JQ4W 44569889 Ki = 3700 nM T17758 CE1O4I 44569890 Ki = 11000 nM T17758 C4JU7I 44569891 Ki = 6200 nM T17758 CGS83Z 44569892 Ki = 3600 nM T17758 C4BN3H 44573109 Ki = 3300 nM T17758 COR57Y 44573272 Ki = 3000 nM T17758 C6DX3Y 44573273 Ki = 2200 nM T17758 CM2R1P 44573274 Ki = 16900 nM T17758 CSP1I0 44573310 Ki = 8370 nM T17758 C6EG9V 44573311 Ki = 7300 nM T17758 CYV3X2 44573378 Ki = 34500 nM T17758 CWUA41 44573379 Ki = 76000 nM T17758 CYA64G 44573380 Ki = 126000 nM T17758 CLG42S 44573428 Ki = 193000 nM T17758 CDW2M8 44574895 IC50 = 16000 nM T17758 C8XT1U 44626341 IC50 = 25 nM T17758 C27ALM 44626342 IC50 > 30000 nM T17758 C7JP5Q 44626343 IC50 = 39 nM T17758 CDG17C 44626344 IC50 = 23 nM T17758 C6I0TN 44626345 IC50 = 15 nM T17758 CUK2I7 45103480 Ki = 120 nM T17758 CP6SB1 45103481 Ki = 170 nM T17758 CM16YW 45103482 Ki = 140 nM T17758 C2PVE0 45103523 Ki > 26000 nM T17758 CKN2F4 45103582 Ki = 190 nM T17758 C80DXA 45103583 Ki = 130 nM T17758 CG51EA 45103584 Ki = 220 nM T17758 C46JPW 45103585 Ki = 310 nM T17758 C8XBZ6 45103586 Ki = 85 nM T17758 CXS6K8 45103587 Ki = 297 nM T17758 CPR1O7 45103680 Ki = 833 nM T17758 CJU8M5 45103681 Ki = 58 nM T17758 CGN14R 45103723 Ki > 26000 nM T17758 CF2DG4 45266265 Ki = 500000 nM T17758 C94RXO 45266266 Ki = 90000 nM T17758 C76JPC 45266296 Ki = 41000 nM T17758 CE20SM 45266980 Ki = 10000 nM T17758 CTDO14 45267035 Ki = 39.81 nM T17758 CJSM84 45267041 Ki = 7943.28 nM T17758 C2CS1D 45267821 Ki = 251.19 nM T17758 CMAN30 45267826 Ki = 3981.07 nM T17758 CY72GK 45267842 Ki = 6309.57 nM T17758 C4ZWL1 45268708 Ki = 630.96 nM T17758 CV4B0J 45268714 Ki = 398.11 nM T17758 CR79DU 45269565 Ki = 10000 nM T17758 C8CL4R 45269570 Ki = 1.585 nM T17758 C6WG8P 45269579 Ki = 31.62 nM T17758 CB94WC 45270387 Ki = 5011.87 nM T17758 CBI54K 45270388 Ki = 15848.93 nM T17758 C1QNL2 45270410 Ki = 1258.93 nM T17758 CMIT36 45270413 Ki = 10000 nM T17758 CVLU57 45270415 Ki = 316.23 nM T17758 C9S8FX 45271213 Ki = 5011.87 nM T17758 C96ATQ 45271222 Ki = 1584.89 nM T17758 C59DXE 45271223 Ki = 398.11 nM T17758 CBC23Z 45271232 Ki = 10000 nM T17758 CQO9K8 45271235 Ki = 3162.28 nM T17758 CCW0D3 45271239 Ki = 3981.07 nM T17758 C4EOK3 45271242 Ki = 5011.87 nM T17758 C6SFK1 45272122 Ki = 39810.72 nM T17758 CDL7Z3 45272132 Ki = 31622.78 nM T17758 CYC70O 45272136 Ki = 10000 nM T17758 CI4MP3 45272948 Ki = 1000 nM T17758 C0X1OF 45272962 Ki = 158.49 nM T17758 CGXD19 45485586 IC50 = 98 nM T17758 C9OZ8H 45485587 IC50 = 100 nM T17758 C5J8QY 45485588 IC50 = 13000 nM T17758 C6RGL9 45485591 IC50 > 30000 nM T17758 C0H5ST 45485592 IC50 = 220 nM T17758 CRJ02S 45485601 IC50 = 26000 nM T17758 CJZ3G7 45485602 IC50 = 3500 nM T17758 C6RA5X 45485603 IC50 = 1300 nM T17758 CY5P2K 45485610 IC50 > 30000 nM T17758 CPT2Y1 45485611 IC50 = 89 nM T17758 CA2WK7 45485615 IC50 > 30000 nM T17758 C27HKO 45485622 IC50 = 240 nM T17758 CF39BN 45485632 IC50 = 2700 nM T17758 C3HKP7 45485641 IC50 = 130 nM T17758 C62BQW 45485647 IC50 = 540 nM T17758 C7UK5D 45485655 IC50 = 680 nM T17758 CHT06J 45485667 IC50 = 530 nM T17758 C76CDZ 45485668 IC50 = 900 nM T17758 CGX93B 45485669 IC50 = 65 nM T17758 C0R4EB 45485670 IC50 = 100 nM T17758 CI5EJ4 45485671 IC50 = 840 nM T17758 CI0V3Q 45485678 IC50 = 20000 nM T17758 CY0P2W 45485679 IC50 > 30000 nM T17758 C10DVP 45485688 IC50 = 8100 nM T17758 C4M1RE 45485689 IC50 > 30000 nM T17758 C9L1ZS 46233075 Ki = 109 nM T17758 CD62VO 46233076 Ki = 251 nM T17758 C5PI6E 46233077 Ki = 59 nM T17758 C9BLH7 46233114 Ki = 156 nM T17758 C42DOH 46233115 Ki = 151 nM T17758 CA7S2F 46233116 Ki = 2115 nM T17758 CQ4UF5 46233117 Ki = 828 nM T17758 CEU41B 46233150 Ki = 940 nM T17758 CXV4P6 46233151 Ki = 650 nM T17758 CHF45Z 46233364 Ki = 2270 nM T17758 CLHX82 46233406 Ki = 500 nM T17758 C8T5CW 46233408 Ki = 2130 nM T17758 CQ01MF 46233409 Ki = 140 nM T17758 CY92TG 46233410 Ki = 510 nM T17758 CT5MH6 46233491 Ki = 160 nM T17758 CY5C1O 46233492 Ki = 270 nM T17758 C5H2EF 46233511 Ki = 250 nM T17758 CZ46CU 46233512 Ki = 140 nM T17758 CI8NV4 46233513 Ki = 210 nM T17758 C84HTG 46233514 Ki = 150 nM T17758 CA4Z5X 46233537 Ki = 440 nM T17758 C5SK7C 46233538 Ki = 510 nM T17758 C0Y8IT 46233539 Ki = 331 nM T17758 C16IMD 46233540 Ki = 935 nM T17758 CW3S0U 46233565 Ki = 780 nM T17758 C03TRU 46233566 Ki = 308 nM T17758 C8RCY2 46233567 Ki = 226 nM T17758 CHO28I 46233568 Ki = 89 nM T17758 CRDC20 46233603 Ki = 1631 nM T17758 CWVY84 46233604 Ki = 201 nM T17758 C7ZP4M 46233605 Ki = 201 nM T17758 CT84CW 46233649 Ki = 308 nM T17758 CF8Z3Q 46233651 Ki = 609 nM T17758 CX28UI 46233688 Ki = 575 nM T17758 C9P0FC 46233689 Ki = 249 nM T17758 CWO0V7 46233690 Ki = 142 nM T17758 C7ET8Q 46233691 Ki = 169 nM T17758 CXUM36 49820499 Ki > 10000 nM T17758 CX7SA8 49820500 Ki > 10000 nM T17758 CQ3R6L 49820501 Ki > 10000 nM T17758 CSFD83 49820654 Ki > 10000 nM T17758 CS8FY6 49820655 Ki = 10 nM T17758 C6OIW8 49820657 Ki > 10000 nM T17758 CJ5G9Q 49820816 Ki = 4 nM T17758 CL8UV3 49820969 Ki = 5 nM T17758 C2B5EC 49820973 Ki = 15 nM T17758 C41JHG 52941953 Ki = 6700 nM T17758 CJ7RF0 52945600 Ki = 400 nM T17758 CA6GQ5 53341037 Ki > 15100 nM T17758 CCR6H5 53357861 IC50 = 1200 nM T17758 CI9GP5 53357862 IC50 = 870 nM T17758 C52ZET 53357863 IC50 = 6300 nM T17758 C53JUT 53357864 IC50 = 10000 nM T17758 C9YK0S 53357865 IC50 = 14000 nM T17758 CV60BK 53488415 Ki = 15100 nM T17758 C8U4OD 56649692 IC50 > 1000000 nM T17758 CZS51B 56663151 IC50 = 12000 nM T17758 CNV1L2 56935636 IC50 = 6000 nM T17758 C9LQF8 56935648 IC50 = 6000 nM T17758 CLU95A 57325502 IC50 = 2800 nM T17758 CKV1M9 57390790 IC50 = 19000 nM T17758 CC32NR 57390791 IC50 = 6900 nM T17758 CV42AN 57390824 IC50 = 4000 nM T17758 C1GIV7 57390825 IC50 = 2600 nM T17758 CX9QT2 57390826 IC50 = 16000 nM T17758 CMY2W6 57390827 IC50 = 31000 nM T17758 C16YVS 57390877 IC50 > 62000 nM T17758 CR1CP9 57390878 IC50 = 30000 nM T17758 CM7FT5 57390879 IC50 = 3600 nM T17758 C73CPY 57390905 IC50 = 14000 nM T17758 C50HMB 57390907 IC50 = 21000 nM T17758 CT8N4P 57391010 IC50 > 222000 nM T17758 CGLI02 57392603 IC50 = 16000 nM T17758 CBTW51 57392644 IC50 = 9000 nM T17758 CMAT35 57392645 IC50 = 12000 nM T17758 C0MK4Y 57392646 IC50 = 31000 nM T17758 C3V2RP 57392647 IC50 = 31000 nM T17758 C3NP4M 57392705 IC50 = 16000 nM T17758 C7UVI1 57392707 IC50 = 61000 nM T17758 CA80YK 57392794 IC50 = 26000 nM T17758 CH75KT 57392806 IC50 = 1000000 nM T17758 CDC12Z 57393288 IC50 > 62000 nM T17758 C3J1OW 57394321 IC50 = 23000 nM T17758 CXV4U9 57394359 IC50 = 2400 nM T17758 C40DMP 57394421 IC50 = 6000 nM T17758 C9LVB6 57394423 IC50 = 15000 nM T17758 CYQ9U4 57394426 IC50 = 43000 nM T17758 CCBI40 57394516 IC50 = 120000 nM T17758 C8H3SV 57396080 IC50 > 62000 nM T17758 CS3R1O 57396081 IC50 = 8000 nM T17758 C06CKD 57396112 IC50 = 8100 nM T17758 C4ZE7U 57396113 IC50 = 11000 nM T17758 C05FIW 57396161 IC50 = 45000 nM T17758 CRC1E9 57396185 IC50 > 1000000 nM T17758 CH2KN8 57396188 IC50 = 15000 nM T17758 C9JCN3 57396267 IC50 = 102000 nM T17758 CN9GI3 57396269 IC50 > 1000000 nM T17758 CIC2U6 57397927 IC50 = 2900 nM T17758 C98KRU 57397928 IC50 = 6400 nM T17758 CI89BC 57397929 IC50 = 7000 nM T17758 C2WMK9 57397993 IC50 > 1000000 nM T17758 CNF64Q 57397995 IC50 = 50000 nM T17758 C1CHI3 57397997 IC50 = 28000 nM T17758 CJI9G2 57398072 IC50 = 37000 nM T17758 C9JMZ7 57399538 IC50 > 62000 nM T17758 C7L0DK 57399539 IC50 > 62000 nM T17758 C72ERX 57399571 IC50 = 20000 nM T17758 C5V1XZ 57399617 IC50 = 15000 nM T17758 CK0M9X 57399649 IC50 = 8000 nM T17758 CIH17N 57399651 IC50 = 6000 nM T17758 C2D7FP 57399653 Ki = 2498 nM T17758 CM9L7G 57399729 IC50 = 44000 nM T17758 C54QWO 57400206 IC50 > 62000 nM T17758 CBKD41 57400356 IC50 = 4100 nM T17758 C3DY5T 57401325 IC50 = 14000 nM T17758 C67MDP 57401326 IC50 > 250000 nM T17758 CKV6R8 57401327 IC50 = 2100 nM T17758 CT0D4V 57401328 IC50 > 31000 nM T17758 CVS3G4 57401380 IC50 = 9800 nM T17758 CCVI24 57401401 IC50 = 10000 nM T17758 C41GJN 57401403 IC50 = 177000 nM T17758 C7ORW9 57401405 IC50 = 3000 nM T17758 CE3C2H 57401407 IC50 = 35000 nM T17758 CNO46U 57401490 IC50 > 1000000 nM T17758 CC09DX 57401495 IC50 > 1000000 nM T17758 CY8UF5 57402007 IC50 > 62000 nM T17758 CNX6O7 57403048 IC50 = 62000 nM T17758 CAYH90 57403049 IC50 = 8000 nM T17758 CES6D2 57403083 IC50 = 4000 nM T17758 C2DL6W 57403084 IC50 = 9800 nM T17758 C0E4FU 57403085 IC50 = 31000 nM T17758 C1J8GI 57403129 IC50 = 16000 nM T17758 CB36VU 57403154 IC50 = 38000 nM T17758 C94BHY 57403156 IC50 = 17000 nM T17758 CX81NW 57403157 IC50 = 30000 nM T17758 C1RS7P 57403239 IC50 > 1000000 nM T17758 CL2ZI5 57403241 IC50 = 25000 nM T17758 C3RZ8G 57404502 IC50 = 4000 nM T17758 CVWP51 57404503 IC50 = 3000 nM T17758 C9XW1C 57842830 Ki > 10000 nM T17758 C60HCV 57976401 Ki > 15100 nM T17758 CHB27Y 57976410 Ki > 29730 nM T17758 CSC0L5 59020200 Ki > 13000 nM T17758 C91APY 59095797 IC50 > 33000 nM T17758 C69SED 59095888 IC50 = 31500 nM T17758 CPW2H7 59315536 Ki > 10000 nM T17758 CO38AC 59402011 Ki > 28000 nM T17758 CE5A7B 60162406 Ki = 8900 nM T17758 CWOD93 66744646 Ki = 5050 nM T17758 CSAQ19 66818162 Ki > 10000 nM T17758 COAY94 66818433 Ki = 13 nM T17758 CG9UM3 66818450 Ki = 9 nM T17758 CSI0K8 66818456 Ki = 12 nM T17758 CG0TZ3 66818504 Ki = 10 nM T17758 CU6E0A 66818541 Ki = 23 nM T17758 C89BXR 66818555 Ki > 10000 nM T17758 C6LD2R 66818559 Ki = 7 nM T17758 C6CP8D 66818568 Ki = 11 nM T17758 CKD8I1 66818569 Ki = 14 nM T17758 C05LHZ 66818575 Ki = 9 nM T17758 CDA2M4 66818582 Ki = 4 nM T17758 C9LTK3 66818589 Ki > 10000 nM T17758 C9FQY8 66818629 Ki = 5 nM T17758 C9GM3F 66818639 Ki = 23 nM T17758 C4U7SZ 66818677 Ki = 12 nM T17758 CL8D0V 66818717 Ki = 17 nM T17758 C41RKZ 66818743 Ki > 10000 nM T17758 C6Q8FO 66818744 Ki = 13 nM T17758 CE53KG 66818763 Ki = 22 nM T17758 CJA30C 66818765 Ki = 9 nM T17758 C5LU1Z 66818766 Ki = 25 nM T17758 CR94HZ 66818781 Ki = 6 nM T17758 CP18VA 66818813 Ki = 19 nM T17758 CF4PT6 66818819 Ki = 1 nM T17758 CYB76J 66818882 Ki = 2 nM T17758 CRH5O7 66818889 Ki > 10000 nM T17758 CGI6B3 66819113 Ki = 9 nM T17758 C4JV1L 66820910 Ki = 12 nM T17758 C62LDA 66821311 Ki = 4 nM T17758 CK59IZ 68788696 Ki = 13 nM T17758 CGA3T2 68789018 Ki = 11 nM T17758 CC0J3V 68790735 Ki = 15 nM T17758 C2B4HJ 69496391 IC50 = 3280 nM T17758 CPY6J2 69496521 IC50 = 360 nM T17758 CPO6Z9 69496614 IC50 = 23 nM T17758 C1DUV4 69496716 IC50 = 7260 nM T17758 C6YW5E 69496717 IC50 = 51 nM T17758 CUG9Z7 69496724 IC50 = 84 nM T17758 CR59OP 69496744 IC50 = 237 nM T17758 CX97VL 69496820 IC50 = 79 nM T17758 CD5ZW0 69496838 IC50 = 34 nM T17758 C6AU1R 70252985 Ki > 29730 nM T17758 CTO5I6 70253788 Ki > 29730 nM T17758 CL4RK8 70683232 IC50 = 212000 nM T17758 CX0VK6 70689516 IC50 = 69000 nM T17758 C2UOG4 70693724 IC50 = 237000 nM T17758 CE27BR 70695842 IC50 = 47000 nM T17758 C9EL3C 71260387 Ki > 15100 nM T17758 CJPF90 71548883 Ki > 15000 nM T17758 C30ZKJ 71561420 Ki = 6500 nM T17758 C62ZTJ 71660643 IC50 > 33000 nM T17758 C78DJQ 71711730 IC50 < 10000 nM T17758 CD53RA 71716975 Ki > 120000 nM T17758 CSP5T2 71716976 Ki > 120000 nM T17758 C5RSD4 71818404 IC50 = 310 nM T17758 CVPL10 71818549 IC50 = 6600 nM T17758 CVCM38 71818688 IC50 = 620 nM T17758 CA56TS 71818689 IC50 = 440 nM T17758 CK2XH0 71818692 IC50 = 1500 nM T17758 CXV8Z4 71818829 IC50 = 480 nM T17758 C7UY4N 71818830 IC50 = 25300 nM T17758 C6X2FC 71818831 IC50 = 13700 nM T17758 C80YBP 71818832 IC50 = 14800 nM T17758 CM83VP 72163524 IC50 > 10000 nM T17758 CRBH34 72164200 IC50 > 33000 nM T17758 CWNZ45 72164201 IC50 > 33000 nM T17758 CLI36U 72551247 Ki = 15000 nM T17758 C1MBU7 72793747 IC50 > 50000 nM T17758 C6BY5D 72793776 IC50 > 50000 nM T17758 C1DI8A 72793778 IC50 > 50000 nM T17758 CAJ7O5 73350148 Ki = 22000 nM T17758 C5U9CI 73355715 Ki = 0.0086 nM T17758 C5MVT3 76310068 Ki > 10000 nM T17758 CFEZ96 76314786 Ki = 4770 nM T17758 C6MK0I 76318385 Ki = 14800 nM T17758 CWZA05 76320988 Ki > 10000 nM T17758 CK9UQ1 76322063 Ki = 710 nM T17758 C35YPH 76329253 Ki = 8670 nM T17758 CN48KP 76329254 Ki = 48700 nM T17758 CV8R1U 76336512 Ki = 900 nM T17758 CJM75B 76336513 Ki = 26800 nM T17758 C8Z4VP 76336514 Ki = 23500 nM T17758 C4G3KH 76336515 Ki = 1480 nM T17758 C5CX4Z 76849444 IC50 > 500000 nM T17758 C9ASZ2 86302628 IC50 > 400000 nM T17758 CMD5V7 86583041 Ki > 14060 nM T17758 CV7IW5 87167024 Ki = 8 nM T17758 CWP85J 87360663 IC50 = 19800 nM T17758 CO6U9I 88582319 Ki > 29730 nM T17758 CJ6CN0 90644019 Ki = 20 nM T17758 CB8KY3 90644020 Ki = 16 nM T17758 C0G6SP 90644022 Ki = 13 nM T17758 CH3US6 90644023 Ki = 15 nM T17758 C9A7YX 90655485 IC50 > 1000000 nM T17758 C90UNY 90655486 IC50 > 200000 nM T17758 C75WHK 90655487 IC50 > 1000000 nM T17758 CZ1Q2P 90655488 IC50 > 1000000 nM T17758 CSG0L5 90655489 IC50 > 400000 nM T17758 C8KX5F 90655490 IC50 > 1000000 nM T17758 C9W1CO 90655491 IC50 > 1000000 nM T17758 C5WIF7 90655492 IC50 > 1000000 nM T17758 C6FE2K 90655493 IC50 > 1000000 nM T17758 C2I7SQ 90655494 IC50 > 1000000 nM T17758 CXY0I6 90655495 IC50 > 1000000 nM T17758 CWL8U1 90655496 IC50 > 1000000 nM T17758 CRQ6I4 90655497 IC50 > 1000000 nM T17758 CL27GQ 90655498 IC50 > 400000 nM T17758 CLG8M0 90655499 IC50 > 1000000 nM T17758 CBK7Y9 90655500 IC50 > 400000 nM T17758 CD7WM6 90655501 IC50 > 1000000 nM T17758 CJ7B8Y 90655502 IC50 > 1000000 nM T17758 CW6VS9 90655503 IC50 > 1000000 nM T17758 CV1NM4 90655504 IC50 > 1000000 nM T17758 CKPN23 90655505 IC50 > 200000 nM T17758 CZ8S4C 90655506 IC50 > 1000000 nM T17758 CI3AX1 90666144 Ki = 4400 nM T17758 C43YWM 90666145 Ki = 3400 nM T17758 CT45NA 90666146 Ki = 18500 nM T17758 C56KQL 90666147 Ki = 18100 nM T17758 CZ0UR6 92220134 IC50 = 285 nM T17758 C65TLW 101862198 Ki > 1000000 nM T17758 CL8WC6 117819668 IC50 > 30000 nM T17758 C2RXZ3 117820231 IC50 = 770 nM T17758 CMJ8R1 118601604 Ki = 28 nM T17758 C0GRU4 118718129 Ki = 81 nM T17758 CHQ5P7 118987013 Ki > 14060 nM T17758 C3NK4O 121232387 Ki = 1300 nM T17758 CTPA56 122179839 IC50 > 200000 nM T17758 CY51OU 122179842 IC50 > 200000 nM T17758 CB8K4S 122179843 IC50 > 200000 nM T17758 CLDC14 122194710 Ki = 2300 nM T17758 C6NGM7 122194711 Ki = 2700 nM T17758 CR4CY8 122194712 Ki = 7800 nM T17758 CFD89O 127021019 IC50 = 77000 nM T17758 CB9V3Y 127025119 IC50 > 100000 nM T17758 CK0W2P 127027635 Ki > 15000 nM T17758 CJ6DA9 127028140 IC50 = 1400 nM T17758 CD9KI3 127028141 IC50 = 7.9 nM T17758 CPC0M8 127031390 Ki > 14060 nM T17758 C3XD2I 127035151 IC50 > 50000 nM T17758 C1BWV2 127035672 Ki > 1000000 nM T17758 CTMR64 127035685 Ki > 1000000 nM T17758 COG73V 127035809 IC50 > 100000 nM T17758 C07FSI 127035810 IC50 > 100000 nM T17758 C73SHP 127035840 IC50 > 100000 nM T17758 CBJ14T 127035841 IC50 > 100000 nM T17758 CM34NK 127035842 IC50 > 200000 nM T17758 C6TS0X 127035843 IC50 > 50000 nM T17758 C6W4AT 127035844 IC50 > 50000 nM T17758 CL6HJ1 127036010 IC50 > 200000 nM T17758 CFWR36 127036011 IC50 > 100000 nM T17758 CHQ42U 127036012 IC50 > 100000 nM T17758 CVRY56 127036086 Ki > 1000000 nM T17758 C54OHE 127036643 IC50 > 100000 nM T17758 CJ0L7S 127036644 IC50 > 100000 nM T17758 CN42TJ 127036645 IC50 > 100000 nM T17758 C76FJU 127036847 IC50 > 100000 nM T17758 CK40VA 127036848 IC50 > 100000 nM T17758 C9B6LT 127037264 Ki > 1000000 nM T17758 C60HLK 127037469 Ki = 93000 nM T17758 C64FQM 127037562 IC50 = 62000 nM T17758 CDBR37 127037804 IC50 = 184 nM T17758 CF07ZO 127037805 IC50 = 254 nM T17758 CU87YF 127037806 IC50 = 174 nM T17758 CN4U9B 127037807 IC50 = 366 nM T17758 C7N0EM 127037808 IC50 = 404 nM T17758 CCS4I9 127039388 IC50 = 9300 nM T17758 C82RFB 127039699 IC50 = 150000 nM T17758 CSB59A 127039709 IC50 = 9040 nM T17758 CF2W3O 127040526 IC50 = 250000 nM T17758 CM0F8N 127040527 IC50 = 19390 nM T17758 CU35ZD 127040830 IC50 > 1000000 nM T17758 C7LVM8 127040831 IC50 = 500000 nM T17758 C0H4VS 127040832 IC50 = 250000 nM T17758 CSV1W9 127040833 IC50 = 63920 nM T17758 CW14DT 127040834 IC50 = 30250 nM T17758 C9A4BF 127040835 IC50 = 48470 nM T17758 C5U6JT 127040836 IC50 = 250000 nM T17758 CA0M2S 127040837 IC50 = 99160 nM T17758 C0CZI3 127041062 IC50 = 500000 nM T17758 CH3V9O 127041159 IC50 = 30150 nM T17758 C9NT1F 127041160 IC50 = 100000 nM T17758 CC53FU 127041161 IC50 = 125000 nM T17758 C8R5QV 127041162 IC50 = 53780 nM T17758 CI9QN2 127041163 IC50 = 27440 nM T17758 CNER57 127041164 IC50 = 14950 nM T17758 CN1VP7 127041165 IC50 = 26850 nM T17758 C8R1WX 127041381 IC50 = 200000 nM T17758 C5JKF6 127041466 IC50 = 6890 nM T17758 C6JGI5 127041467 IC50 = 23890 nM T17758 C96JWU 127041468 IC50 = 200000 nM T17758 C46BAW 127041469 IC50 = 57550 nM T17758 CYZ43P 127041470 IC50 = 60840 nM T17758 CO24MD 127041471 IC50 = 27260 nM T17758 C85ROH 127041472 IC50 = 97 nM T17758 CPX74M 127041993 IC50 = 18030 nM T17758 C8MKE9 127045985 IC50 = 160000 nM T17758 C6T3JF 127045986 IC50 > 200000 nM T17758 CV4TI5 127045987 IC50 > 200000 nM T17758 CK6D1Z 127045988 IC50 > 200000 nM T17758 C3ZP4A 127046388 IC50 > 200000 nM T17758 C8IVS0 127046389 IC50 > 200000 nM T17758 CBL5K4 127046390 IC50 > 200000 nM T17758 C6TYG9 127046555 IC50 > 200000 nM T17758 CHDW47 127046556 IC50 > 200000 nM T17758 C21JMT 127046792 IC50 = 150000 nM T17758 CN2M8P 134154823 Ki = 53 nM T17758 C6HTD5 135393470 Ki = 183 nM T17758 COZ79Q 135393472 Ki = 166 nM T17758 C7NA6E 135393474 IC50 = 39 nM T17758 CY4VK1 135393475 Ki = 42 nM T17758 C5XA6H 135407717 Ki = 3600 nM T17758 C0OX6T 135407736 Ki = 3300 nM T17758 C61XOA 135427245 Ki = 3600 nM T17758 C8WS4O 135443730 Ki = 7500 nM T17758 CTP5V8 135444609 Ki = 400 nM T17758 C4M5BF 135450980 Ki = 2000 nM T17758 CXS6B9 135471524 Ki = 1900 nM T17758 C2PFI8 135475618 Ki = 900 nM T17758 CBE9G0 135490854 Ki = 3900 nM T17758 CMQ6O0 135501618 Ki = 8000 nM T17758 CVA61N 135512760 Ki = 3700 nM T17758 CK97FT 135533257 Ki = 500 nM T17758 CAD75F 135535997 Ki = 11000 nM T17758 CCH49A 135544551 Ki = 550 nM T17758 CKLD47 135544579 Ki = 13000 nM T17758 CQD2Z1 135855944 Ki = 0.46 nM T17758 C9G7TE 135995982 Ki = 550 nM T17758 C6S5OL 136034781 Ki = 1200 nM T17758 CN70IU 136092208 Ki = 950 nM T17758 C5N3KP 136092209 Ki = 100 nM T17758 C1BUH6 136092210 Ki = 460 nM T17758 CFQ2C8 136092211 Ki = 180 nM T17758 CX5R9J 136092212 Ki = 110 nM T17758 C35PXN 136092213 Ki = 220 nM T17758 CEXJ30 136092214 Ki = 290 nM T17758 CS6QH0 136092215 Ki = 550 nM T17758 CMR7L4 136092216 Ki = 700 nM T17758 CN0WR7 136092217 Ki = 80 nM T17758 COCN35 136092218 Ki = 32 nM T17758 CA79JC 136092219 Ki = 700 nM T17758 C26ZPI 136264091 IC50 = 279000 nM T17758 C8VJW4 136266885 IC50 = 74000 nM T17758 CC0BI4 136268735 IC50 = 231000 nM T17758 CYP96F 137348032 Ki = 508 nM T17758 CV3QJ5 137348787 Ki = 108 nM T17758 CX7V8Y 137349240 Ki = 156 nM T17758 CUZ35A 138115400 IC50 > 100000 nM T17758 CD7Y4N 138810990 Ki = 482 nM T17758 C41EJL 139030450 Ki = 204 nM T17758 CL5ES9 139030451 Ki = 1626 nM T17758 CO51HN 139030452 Ki = 302 nM T17758 CX07YE 139592452 Ki > 15100 nM T17758 CRE5O9 145960395 IC50 = 58000 nM T17758 C0M2QA 145960406 IC50 = 1000 nM T17758 CRK0L6 145960477 IC50 > 14000 nM T17758 C0OF9H 145960548 IC50 = 24500 nM T17758 C36PYJ 145960730 IC50 = 22000 nM T17758 CW9X7P 145960760 IC50 = 140000 nM T17758 C47IGD 145960856 IC50 = 64000 nM T17758 CXI16W 145960913 IC50 = 60000 nM T17758 C41LXH 145960914 IC50 = 2430 nM T17758 C02KUI 145961020 IC50 = 12000 nM T17758 CK7H3W 145961084 IC50 = 4700 nM T17758 C25NZG 145961305 IC50 = 8000 nM T17758 CG6R0N 145961689 IC50 = 18000 nM T17758 CXUW40 145961875 IC50 = 24000 nM T17758 CD0I6N 145962360 IC50 = 68000 nM T17758 CGV68W 145962449 IC50 = 11000 nM T17758 COXY65 145962472 IC50 = 4400 nM T17758 C39NWG 145962609 IC50 = 43000 nM T17758 CZN4A5 145962690 IC50 > 19000 nM T17758 CJ6Y4W 145962813 IC50 = 3000 nM T17758 CR78WU 145963185 IC50 = 19000 nM T17758 C93BRK 145963190 IC50 = 5300 nM T17758 CD31BO 145963222 IC50 = 16000 nM T17758 CA8J7F 145963231 IC50 = 7200 nM T17758 CE6C0A 145970642 Ki = 13330 nM T17758 CMSJ87 146029516 Ki = 1778 nM T17758 C8VLB4 146029517 Ki = 1319 nM T17758 CX6C2H 146029518 Ki = 4255 nM T17758 C0VD6T 146029519 Ki = 43 nM T17758 C2VGQ8 146029520 Ki = 1027 nM T17758 CN46IC 146029521 Ki = 228 nM T17758 CG62QA 146029522 Ki = 3308 nM T17758 C4HLX8 146029523 Ki = 88 nM T17758 C6MS5U 146033827 Ki = 884 nM T17758 C6J4QT 146033828 Ki = 5670 nM T17758 CXMU86 146033829 Ki = 42 nM T17758 C2B7TI 146033831 Ki = 41 nM T17758 CA5B4F 146033832 Ki = 315 nM T17758 CP40NR 146033833 Ki = 2417 nM T17758 C4FL0W 146033834 Ki = 658 nM T17758 C1CIF7 146033835 Ki = 21 nM T17758 CDX9J7 146034186 Ki = 16441 nM T17758 CCV3M4 146034187 Ki = 2198 nM T17758 CS6Q0Z 146034188 Ki = 934 nM T17758 C4Q3GP 146034879 Ki = 3539 nM T17758 CICU31 155511394 Ki = 2033 nM T17758 CZR36C 155511554 IC50 = 79432.82 nM T17758 C2VX3G 155512946 Ki > 15100 nM T17758 C71YDF 155513178 Ki = 499 nM T17758 C2CI8S 155513907 Ki = 4435 nM T17758 CYT20V 155514020 Ki > 50000 nM T17758 CAT98N 155514640 Ki > 10000 nM T17758 C4GCY9 155518047 Ki = 287 nM T17758 CF96DM 155518671 Ki > 10000 nM T17758 COFN28 155519549 Ki = 587 nM T17758 C6NX4K 155519661 IC50 = 12589.25 nM T17758 C4MS1B 155519676 IC50 > 100000 nM T17758 CD26NE 155520905 Ki = 3136 nM T17758 C7DUX3 155520916 Ki > 10000 nM T17758 C0EUP5 155521416 Ki = 776 nM T17758 CO7UX6 155522078 Ki = 771 nM T17758 CN3BH5 155527998 IC50 = 5011.87 nM T17758 CHYW65 155528639 IC50 = 79432.82 nM T17758 CD7O2G 155530095 IC50 > 100000 nM T17758 C46AZL 155530642 Ki = 340 nM T17758 C35QWO 155531023 IC50 > 100000 nM T17758 C12HON 155536142 IC50 > 100000 nM T17758 C1KUA7 155538532 Ki = 1208 nM T17758 CL90DN 155540666 Ki > 10000 nM T17758 CY6DK3 155540964 IC50 = 63.1 nM T17758 C4P2GV 155543617 Ki = 15000 nM T17758 C40BTW 155544256 Ki = 904 nM T17758 C5MB9R 155547962 IC50 = 50118.72 nM T17758 CLFB25 155548371 IC50 > 100000 nM T17758 CU9FL4 155551858 Ki > 50000 nM T17758 COM52R 155551892 IC50 = 79432.82 nM T17758 C28ESB 155552505 Ki = 439 nM T17758 CHDB63 155553525 Ki = 1414 nM T17758 CJ3FI5 155553630 IC50 > 100000 nM T17758 CI6SF0 155553995 Ki = 1259 nM T17758 C8JRK9 155554981 Ki = 1477 nM T17758 C0ZR2J 155555188 Ki = 350 nM T17758 CU8LR3 155555208 Ki = 903 nM T17758 CZ8NH9 155556228 Ki = 578 nM T17758 CSW48V 155557718 IC50 = 7943.28 nM T17758 CV7OE8 155560933 Ki = 642 nM T17758 CYA90F 155562662 Ki = 3645 nM T17758 CM8XB1 155565537 IC50 = 50118.72 nM T17758 CP4F1U 155567613 Ki > 50000 nM T17758 CEZ8B9 155568406 Ki > 50000 nM T17758 C7L3VJ 155569306 Ki = 2409 nM T17758 CD81GH 46830813 IC50 > 605000 nM T17758 D00PEJ 16658631 Ki = 160 nM T17758 D00POF 21707121 Ki = 1200 nM T17758 D00WFQ 674641 IC50 = 1300 nM T17758 D01JUI 44339119 Ki = 130 nM T17758 D01LCS 447480 Ki = 220 nM T17758 D02AKP 695069 IC50 = 2500 nM T17758 D02AVL 18376720 Ki > 5000 nM T17758 D02NRY 674650 IC50 = 51200 nM T17758 D02PAU 16731825 Ki > 5000 nM T17758 D02XJW 10313318 Ki = 6000 nM T17758 D02YIW 1794 Ki = 1356 nM T17758 D03NLL 180621 IC50 > 1000000 nM T17758 D05DNW 9820186 Ki = 530 nM T17758 D05ZIP 674656 IC50 = 1700 nM T17758 D06AVE 10200844 Ki = 47 nM T17758 D06CJP 16658353 Ki = 140 nM T17758 D06HOI 44249821 Ki > 7800 nM T17758 D06LPR 674651 IC50 = 18200 nM T17758 D06MTX 1506 Ki = 5500 nM T17758 D07PSW 10219978 Ki = 7100 nM T17758 D07SFI 2332 Ki = 180000 nM T17758 D08HOJ 34677 Ki = 39810.72 nM T17758 D08OCL 44331823 Ki > 200000 nM T17758 D08OCS 699665 IC50 = 3100 nM T17758 D08WQJ 700133 IC50 = 47900 nM T17758 D09KKF 162636 IC50 = 200000 nM T17758 D09TNA 44332077 Ki = 24400 nM T17758 D09YLF 44339283 Ki = 4800 nM T17758 D09YQM 9802488 IC50 = 135 nM T17758 D0A8WP 447732 Ki = 630 nM T17758 D0C3QE 21192457 Ki = 4800 nM T17758 D0EH1F 44332057 Ki > 100000 nM T17758 D0F6EZ 44436702 Ki = 16000 nM T17758 D0G4LX 46233650 Ki = 733 nM T17758 D0IU5E 716930 IC50 = 1500 nM T17758 D0J1CC 11948634 Ki > 10000 nM T17758 D0J1QT 44473100 Ki > 7800 nM T17758 D0K0GU 44392430 Ki = 168 nM T17758 D0K4PK 16658352 Ki = 280 nM T17758 D0K7YL 447476 Ki = 8 nM T17758 D0M2PE 29012033 Ki = 191000 nM T17758 D0N1PW 134348 Ki = 25600 nM T17758 D0ON2Z 204102 Ki > 2300 nM T17758 D0P7NY 23661637 IC50 = 50000 nM T17758 D0R9CH 3400921 Ki > 5000 nM T17758 D0S4MQ 44392405 Ki = 820 nM T17758 D0SP2I 6852210 Ki = 1300 nM T17758 D0X1OY 674628 IC50 = 2600 nM T17758 D0Y5IQ 44255320 IC50 = 10000 nM T17758 D0Z7YI 44331573 Ki = 40300 nM T42447 D0E3TC 44259 IC50 = 173 nM T42447 CACS26 11561968 Ki > 10000 nM T42447 CU0E8O 11690457 Ki > 10000 nM T42447 CB0AP2 11705863 Ki > 10000 nM T42447 CV63UL 67240318 IC50 > 10000 nM T49925 D03ZBT 11626560 IC50 > 10000 nM T49925 D04LVK 57379345 IC50 = 1947 nM T49925 D09KTS 24821094 IC50 = 1.82 nM T49925 D0OB0F 5328940 IC50 = 1.1 nM T49925 D0E3TC 44259 IC50 = 1.15 nM T49925 D0G5XV 135565884 IC50 = 155 nM T49925 D0M9QZ 11485656 IC50 = 500000 nM T49925 D0O6VZ 25254071 IC50 = 697 nM T49925 D0T3ME 156422 IC50 = 8500 nM T49925 CVOW82 11238420 IC50 = 37900 nM T49925 CFJ6B2 11441375 IC50 = 396 nM T49925 CE0KI4 11753519 IC50 = 17900 nM T49925 CQG45C 16109001 IC50 = 8300 nM T49925 C1U8XW 16109036 IC50 = 43 nM T49925 CJA0D6 18451024 IC50 = 26500 nM T49925 C6FQB7 18451036 IC50 = 14100 nM T49925 CQNP54 24764449 IC50 = 328 nM T49925 CC71QJ 27666048 IC50 > 100000 nM T49925 C8B6TY 42628503 EC50 < 500 nM T49925 C3VRO9 44557921 IC50 > 10000 nM T49925 C8NA4L 53384644 IC50 > 30000 nM T49925 CV13QY 58540422 IC50 = 1033 nM T49925 CV63UL 67240318 IC50 > 10000 nM T49925 COU73Y 71226944 IC50 = 28 nM T49925 C40JOZ 71235465 IC50 = 69 nM T49925 CDJY72 71568837 IC50 = 1900 nM T49925 C8CAG7 71578921 IC50 > 10000 nM T49925 CZM1K4 71765510 IC50 = 41 nM T49925 C08KEM 122179540 IC50 = 6400 nM T49925 C3AJ4C 122179546 IC50 = 8700 nM T49925 CG0RP7 122179547 IC50 = 2800 nM T49925 C1A0SQ 122179548 IC50 = 5900 nM T49925 C2LAM7 126591927 IC50 = 65 nM T49925 CXC69T 137321158 IC50 = 470 nM T49925 CZOD53 137633880 IC50 = 203 nM T49925 C7BJY5 137636807 IC50 = 39 nM T49925 CO89DX 137649100 IC50 = 22 nM T49925 CINE03 137652514 IC50 = 268 nM T49925 C28QUP 137652864 IC50 = 133.3 nM T49925 C2MD1Q 155513187 IC50 > 10000 nM T49925 C3NA2I 155519537 IC50 = 28 nM T49925 D03OKV 9844320 IC50 > 2.8 nM T49925 D06WGX 9549184 IC50 = 14100 nM T49925 D08RZB 11153014 IC50 < 1 nM T49925 D0E7VO 59627005 IC50 = 2.2 nM T49925 D0L4WN 31420 IC50 = 24000 nM T49925 D0US9O 45275255 IC50 = 33 nM T37735 D0D1SG 5755 EC50 = 32 nM T37735 CR68MZ 6323453 Ki = 850 nM T37735 CYI7T4 9802231 EC50 = 53.7 nM T37735 C59VXD 10386752 EC50 = 14.2 nM T37735 CFVP19 10428095 EC50 = 66 nM T37735 CVQS04 10454813 EC50 = 37.7 nM T37735 CW6P7A 11244720 EC50 = 181.6 nM T37735 CXG0C2 11269006 EC50 = 66 nM T37735 C4SC0W 11281576 EC50 = 129.2 nM T37735 C2WVO7 13877991 Ki = 75000 nM T62998 D0M9GE 53389 IC50 = 1200 nM T62998 CYZ8V2 11786594 IC50 = 100 nM T62998 CEY81K 24968246 IC50 = 79.43 nM T62998 CP65NG 44192214 IC50 = 50 nM T62998 CTR3C2 44193524 IC50 = 50 nM T62998 CHN8Y2 44193611 IC50 = 15 nM T62998 C19RKQ 57393761 IC50 = 1.5 nM T62998 C7IT1S 57397327 IC50 = 630 nM T62998 C5F2JD 57400722 IC50 = 230 nM T62998 C0Z1FJ 57402501 IC50 = 600 nM T62998 C3KJQ7 62705134 IC50 = 50 nM T62998 CE49TA 62705135 IC50 = 1.5 nM T62998 CJ80EC 62705136 IC50 = 50 nM T62998 CNI86V 62705137 IC50 = 15 nM T62998 CTDY10 62705138 IC50 = 1.5 nM T62998 CFI7L6 62705139 IC50 = 1.5 nM T62998 CZ9UX0 62705298 IC50 = 1.5 nM T62998 CX7Q2A 62705299 IC50 = 1.5 nM T62998 CL96NU 62705302 IC50 = 1.5 nM T62998 CM02KZ 62705303 IC50 = 5 nM T62998 CC0P3H 62705467 IC50 = 15 nM T62998 C53CLZ 62705468 IC50 = 1.5 nM T62998 CW7DH3 62705471 IC50 = 1.5 nM T62998 CZ4ON7 62705642 IC50 = 5 nM T62998 CG7KB3 62705643 IC50 = 1.5 nM T62998 C9NOA6 62705646 IC50 = 15 nM T62998 CBO4R7 62705816 IC50 = 15 nM T62998 CU12FX 62707244 IC50 = 10 nM T62998 CS95PE 62707405 IC50 = 30 nM T62998 CTPL64 62707406 IC50 = 500 nM T62998 C4MEN2 62707407 IC50 = 50 nM T62998 C5NP6H 62707409 IC50 = 15 nM T62998 CIV8W1 62707410 IC50 = 50 nM T62998 C39ZAU 62707566 IC50 = 5 nM T62998 CBMS16 62707567 IC50 = 15 nM T62998 C4WF6K 62707568 IC50 = 1.5 nM T62998 CU6HT5 62707569 IC50 = 1.5 nM T62998 C3DZW7 62707570 IC50 = 1.5 nM T62998 C9UO2W 62707571 IC50 = 1.5 nM T62998 C6DF5V 67091351 IC50 = 50.12 nM T62998 CM3SU7 71450129 IC50 = 1.5 nM T62998 CPJ6G3 127031927 IC50 = 39.81 nM T62998 CCLW18 127031928 IC50 = 5011.87 nM T62998 CH3OX5 127032198 IC50 = 50.12 nM T62998 C2G9AO 127032199 IC50 = 158.49 nM T62998 CAN6Q8 127033110 IC50 = 1000 nM T62998 CP57VF 127033111 IC50 = 50.12 nM T62998 CQ05UJ 127033112 IC50 = 50.12 nM T62998 CQ3T1B 127033113 IC50 = 1000 nM T62998 CMUA16 127033389 IC50 = 501.19 nM T62998 CD9ZX0 127033751 IC50 = 199.53 nM T62998 CDXJ29 127034025 IC50 = 158.49 nM T62998 C4DIS0 127034223 IC50 > 31622.78 nM T62998 C9C6QD 127034481 IC50 = 1000 nM T98269 D0J3SU 9847835 EC50 > 5000 nM T98269 D0U6WQ 153270 IC50 = 3.6 nM T98269 D0F9FA 5311139 Ki = 0.7 nM T98269 CV7IN2 104934 Ki = 50 nM T98269 CVX5Z8 644194 Ki = 1700 nM T98269 CT4YC1 5287959 IC50 = 1800 nM T98269 C3T8NF 5288850 IC50 > 20000 nM T98269 CRA84T 5289080 Ki = 5 nM T98269 C3J7CO 5289240 Ki = 120 nM T98269 C1KR5B 5327301 Ki = 12000 nM T98269 C37TKL 5327302 Ki = 160 nM T98269 C64ZMN 5327304 Ki = 3900 nM T98269 C3IZ2W 5327307 Ki = 8300 nM T98269 C16DTL 5327308 Ki = 1900 nM T98269 C4O3QY 5327309 Ki = 3200 nM T98269 C3GUM7 5327310 Ki = 2700 nM T98269 C3LZX9 8027611 IC50 > 25000 nM T98269 CH47VY 9795859 IC50 = 5500 nM T98269 CFN2P6 9800285 Ki = 21000 nM T98269 CE7I9W 9806986 IC50 = 0.13 nM T98269 CYFG94 9807028 IC50 = 6000 nM T98269 CD3P2F 9807170 IC50 = 0.46 nM T98269 C3S1EP 9807375 IC50 = 0.9 nM T98269 C13PRZ 9809421 IC50 = 1600 nM T98269 CDB06Z 9810472 IC50 = 3.4 nM T98269 CLTO67 9821317 IC50 = 20 nM T98269 C4XO3K 9821545 IC50 > 10000 nM T98269 C4W5DI 9827540 IC50 = 2900 nM T98269 CLAC59 9828058 Ki = 48 nM T98269 C6S3KT 9840223 IC50 > 15000 nM T98269 C7C1TN 9845918 Ki = 15 nM T98269 C1MY7K 9848628 Ki = 0.6 nM T98269 CN02PU 9849845 IC50 = 0.67 nM T98269 C5MCX4 9849846 IC50 = 1.08 nM T98269 CDC86G 9850642 IC50 = 1.82 nM T98269 CJO3A5 9851213 IC50 = 0.22 nM T98269 C56LDH 9851279 IC50 = 5450 nM T98269 C6O0QH 9852052 IC50 = 0.31 nM T98269 C2N3LE 9871540 IC50 = 0.99 nM T98269 CX17DM 9871570 IC50 = 1.93 nM T98269 CF0V7B 9871631 IC50 = 0.19 nM T98269 COB39D 9888758 IC50 = 62 nM T98269 CLQH78 9892350 IC50 = 0.92 nM T98269 CW75OE 9892652 IC50 = 0.4 nM T98269 C3YAL4 9895375 IC50 = 1650 nM T98269 C2DMG1 9914167 IC50 > 10000 nM T98269 CK15RJ 9916276 IC50 = 0.087 nM T98269 C0D2IJ 9936767 IC50 = 0.065 nM T98269 CG90WC 9939287 IC50 = 3800 nM T98269 CFCK64 9939773 IC50 = 4200 nM T98269 CN63JG 9958554 IC50 = 0.23 nM T98269 C4RQU8 10000969 Ki = 4800 nM T98269 C9CV0Y 10001828 IC50 = 570 nM T98269 CW4Q3N 10031194 IC50 = 5000 nM T98269 C9Q0BX 10066296 IC50 = 300 nM T98269 CHWA42 10074552 IC50 = 2600 nM T98269 CPBV30 10085754 IC50 = 500 nM T98269 CXB19Y 10248513 Ki = 3500 nM T98269 CMR75W 10318568 IC50 = 900 nM T98269 CLP14S 10322660 Ki = 25 nM T98269 CJ2HB6 10325387 Ki = 2.2 nM T98269 CZ3IH4 10414828 IC50 = 1800 nM T98269 CUX97M 10529912 Ki = 1 nM T98269 CX67SZ 10826725 Ki = 18000 nM T98269 CBK06L 10861643 IC50 > 100000 nM T98269 CDX7A4 10963183 Ki = 25000 nM T98269 C7HSX0 11189577 IC50 = 14 nM T98269 C8BHT1 11402215 Ki = 9600 nM T98269 C4F8DC 11444079 IC50 > 10000 nM T98269 CDT9G3 11467504 IC50 = 0.11 nM T98269 CV4CP9 11496333 IC50 > 10000 nM T98269 CGE2J0 11497112 IC50 > 50000 nM T98269 C6IS9K 11509289 IC50 > 10000 nM T98269 C6L2MY 11509300 IC50 > 5000 nM T98269 CC31QO 11509301 IC50 > 5000 nM T98269 CS8OX7 11510566 IC50 > 10000 nM T98269 C7FY9B 11512139 IC50 > 50000 nM T98269 C15VFG 11515586 IC50 > 25000 nM T98269 CW6PC0 11519268 IC50 > 50000 nM T98269 CZC5D9 11525874 IC50 > 10000 nM T98269 C5BNE1 11533326 IC50 > 50000 nM T98269 CDK3Z5 11533935 IC50 > 10000 nM T98269 C4IC7E 11541867 IC50 > 500000 nM T98269 C3P2GZ 11548424 IC50 > 7000 nM T98269 CVX4M6 11548909 EC50 > 5000 nM T98269 CF0V3P 11576540 IC50 > 10000 nM T98269 C1T9DY 11576622 IC50 > 50000 nM T98269 C03KPR 11576852 EC50 > 5000 nM T98269 CN67DR 11583840 IC50 > 10000 nM T98269 CPD0M8 11584106 IC50 > 50000 nM T98269 CL16IM 11591540 IC50 > 10000 nM T98269 CE2TX6 11591919 IC50 > 15000 nM T98269 CG4Z9A 11598106 IC50 > 10000 nM T98269 C2A4DY 11598117 Ki = 190 nM T98269 CV6MF1 11614728 IC50 > 500000 nM T98269 CFP19E 11619968 IC50 > 50000 nM T98269 CA0LH6 11624920 IC50 > 10000 nM T98269 CEY39D 11628992 IC50 > 500000 nM T98269 C6Y5MG 11634372 IC50 > 10000 nM T98269 CKJE92 11634649 IC50 > 50000 nM T98269 C4QB6F 11635889 IC50 = 1 nM T98269 C2KFU3 11647018 IC50 > 10000 nM T98269 CN32TX 11664423 IC50 > 500000 nM T98269 CUD05C 11670894 IC50 > 50000 nM T98269 CX97NT 11684618 IC50 > 50000 nM T98269 C05YRV 11699954 IC50 > 500000 nM T98269 CKEX64 11700402 IC50 > 500000 nM T98269 C89COT 11705942 IC50 > 10000 nM T98269 C86PAH 11712912 IC50 > 5000 nM T98269 CY90EM 11712953 IC50 = 1 nM T98269 CNV75J 11713799 IC50 19 nM T98269 CJHC37 11744164 Ki = 5 nM T98269 C7QK5F 11755713 IC50 = 28000 nM T98269 CWDK21 11798262 Ki = 1 nM T98269 CM06CE 12085099 IC50 = 5000 nM T98269 CN42BS 12085102 IC50 = 700 nM T98269 CG84MJ 12085104 IC50 > 250000 nM T98269 C5HEB0 12085105 IC50 = 2000 nM T98269 C6T7CV 12085106 IC50 = 2000 nM T98269 C2A0FJ 12085110 IC50 = 66000 nM T98269 C6LKC9 13092389 IC50 > 250000 nM T98269 CJF1L7 13688814 IC50 = 3000 nM T98269 C67COU 14450230 IC50 = 57000 nM T98269 CJ57OA 14585243 Ki = 130 nM T98269 CZ97MI 15384596 Ki = 2700 nM T98269 CZT6E3 15895228 IC50 = 13000 nM T98269 CD85JG 15895230 IC50 = 5000 nM T98269 CX46YB 15931057 Ki = 9 nM T98269 CRWS56 16046172 IC50 = 30 nM T98269 C2BN3P 16215350 IC50 = 5 nM T98269 C7YI1R 16725993 IC50 = 9 nM T98269 CXH9M5 16749067 IC50 = 1830 nM T98269 C2DJ5W 16749068 IC50 > 15000 nM T98269 COM07G 16749069 IC50 = 2825 nM T98269 CPG8Q0 16749161 IC50 = 2300 nM T98269 CG84TK 16749162 IC50 = 3250 nM T98269 CT3HD1 16749163 IC50 = 2720 nM T98269 CZM4X2 16749164 IC50 = 3900 nM T98269 CUZ8N4 16749267 IC50 > 15000 nM T98269 CMEK96 16749268 IC50 > 15000 nM T98269 C01HBN 16749269 IC50 = 6220 nM T98269 CWG3C8 16749270 IC50 = 5700 nM T98269 C8R3GD 16749271 IC50 = 3400 nM T98269 CK2X1Z 17871446 IC50 = 168000 nM T98269 C4CK5U 17871463 Ki = 37000 nM T98269 CH02DX 18354256 Ki = 11000 nM T98269 C8JW0M 18354265 Ki = 65000 nM T98269 C02NJM 18354267 Ki = 22000 nM T98269 CNV18E 18354276 Ki = 16000 nM T98269 CDU6Q9 18354277 Ki = 34500 nM T98269 CI8ZJ5 18354282 Ki = 735000 nM T98269 C70AOM 18354287 Ki = 33000 nM T98269 CFW67Q 22849799 IC50 = 0.76 nM T98269 CB08SP 22875501 IC50 = 2 nM T98269 C59RVP 22881952 Ki = 900 nM T98269 C2Y8BD 22881953 Ki = 3500 nM T98269 CG9TS4 22881956 Ki = 150 nM T98269 COG9A1 22881958 Ki = 1000 nM T98269 C5L1BO 23320791 IC50 = 110000 nM T98269 CM7B5P 23644615 Ki = 11 nM T98269 CW9HL5 23645230 IC50 = 3050 nM T98269 C5G2IL 23645238 IC50 = 1030 nM T98269 C74OPE 23645239 IC50 = 21200 nM T98269 CK7B2A 23645240 IC50 = 4160 nM T98269 C8YA0T 23645241 IC50 = 4060 nM T98269 C8J7UY 23645242 IC50 > 10000 nM T98269 C3MGC1 23645243 IC50 = 3015 nM T98269 CLSU45 23645244 IC50 > 10000 nM T98269 C95KHP 23645245 IC50 = 18900 nM T98269 C08UYG 23645246 IC50 > 10000 nM T98269 C6YEO7 23645247 IC50 > 10000 nM T98269 CFH23D 23645248 IC50 = 18400 nM T98269 CY0M3Z 23645249 IC50 = 9590 nM T98269 C4TIM0 23645250 IC50 > 10000 nM T98269 CZ9HT6 23645253 IC50 = 6190 nM T98269 CZ59CM 23645306 IC50 = 860 nM T98269 CNU1R6 23645307 IC50 = 2600 nM T98269 C8WF2G 23645308 IC50 = 14000 nM T98269 CBSA54 23645309 IC50 = 6500 nM T98269 C9K5WP 24879338 IC50 = 610 nM T98269 CTI80F 25178948 EC50 > 5000 nM T98269 C2GI4J 25178949 EC50 > 5000 nM T98269 CQ2GM9 25178950 EC50 > 5000 nM T98269 C4GFV6 25179140 EC50 > 5000 nM T98269 CYL36B 25179141 EC50 > 5000 nM T98269 CGC69Q 25179143 EC50 > 5000 nM T98269 C27YJF 25179144 EC50 > 5000 nM T98269 C2YTB7 25179145 EC50 > 5000 nM T98269 C6GTV3 25179324 EC50 > 5000 nM T98269 CIC46T 25179513 EC50 > 5000 nM T98269 CK96WB 25179514 EC50 > 5000 nM T98269 CGX78D 25217029 IC50 > 36000 nM T98269 CW2L9Q 25217030 IC50 = 3500 nM T98269 C8UTC4 25217031 IC50 = 2900 nM T98269 CZ43KQ 25217032 IC50 > 10000 nM T98269 C2P9NI 25217145 IC50 > 20000 nM T98269 C8C9XU 42618276 IC50 > 25000 nM T98269 CFO93N 42618277 IC50 > 10000 nM T98269 CS1KQ0 42618278 IC50 = 4100 nM T98269 CVI16X 42618279 IC50 > 10000 nM T98269 C3MRA0 42618280 IC50 > 10000 nM T98269 C8UO9S 42618281 IC50 = 3875 nM T98269 C68NPR 42618282 IC50 = 6825 nM T98269 CL41SD 42618283 IC50 = 5350 nM T98269 CJ7U2E 42618284 IC50 = 4575 nM T98269 CZL8C7 42618285 IC50 = 4300 nM T98269 CNIQ28 42618286 IC50 = 5350 nM T98269 C91OMB 42618287 IC50 > 10000 nM T98269 C5AC1L 42618288 IC50 = 3300 nM T98269 CFU5T2 42618289 IC50 = 4183 nM T98269 CK9H3M 42618290 IC50 > 10000 nM T98269 CV4H2J 42618291 IC50 = 4700 nM T98269 C7VPU3 42618292 IC50 = 4700 nM T98269 C6R2FM 42618293 IC50 > 10000 nM T98269 CL0M7R 44143089 IC50 = 16218.1 nM T98269 C9QDC0 44143091 IC50 = 70794.58 nM T98269 CT7VO2 44157085 IC50 > 500000 nM T98269 CWMU91 44157086 IC50 > 500000 nM T98269 C6LZ5Y 44157087 IC50 > 500000 nM T98269 CYSJ79 44157089 IC50 > 500000 nM T98269 CMX7W1 44157090 IC50 > 500000 nM T98269 C7B3VE 44158086 IC50 > 500000 nM T98269 C20WEJ 44158089 IC50 > 500000 nM T98269 C68KOD 44158154 IC50 > 500000 nM T98269 C4C1RU 44158155 IC50 > 500000 nM T98269 CN1YR9 44158157 IC50 > 500000 nM T98269 C80XPD 44158237 IC50 > 500000 nM T98269 CN09UV 44158238 IC50 > 500000 nM T98269 CT9DF4 44158240 IC50 > 500000 nM T98269 CHDF62 44158242 IC50 > 500000 nM T98269 CS6X1C 44158325 IC50 > 500000 nM T98269 C17TEZ 44158326 IC50 > 500000 nM T98269 CZ0VT3 44158328 IC50 = 3160 nM T98269 C7ERP0 44264266 IC50 > 250000 nM T98269 CJTA60 44264267 IC50 > 250000 nM T98269 CT42GH 44264305 IC50 = 18000 nM T98269 CA4TE9 44264306 IC50 = 5000 nM T98269 CUL19P 44264309 IC50 = 10000 nM T98269 C9W4YO 44264310 IC50 > 250000 nM T98269 C4RKB0 44264332 IC50 = 4000 nM T98269 CM02QP 44264485 IC50 = 1500 nM T98269 CNM4J5 44264544 IC50 > 250000 nM T98269 C74TKQ 44264570 IC50 > 250000 nM T98269 C25EJC 44273962 Ki = 90 nM T98269 CB1N2K 44276330 Ki = 160 nM T98269 CWDE12 44276372 Ki = 14 nM T98269 CGA87O 44276373 Ki = 7 nM T98269 CF3DI4 44276374 Ki = 45 nM T98269 CMLZ84 44276407 Ki = 590 nM T98269 CAPT63 44276436 Ki = 2 nM T98269 COGK42 44276489 Ki = 16 nM T98269 C2UE7W 44276490 Ki = 68 nM T98269 CF8VA9 44276494 Ki = 1.3 nM T98269 C0ES6O 44276495 Ki = 1.8 nM T98269 C6OEI2 44276496 Ki = 1.5 nM T98269 C6JHE1 44276514 Ki = 95 nM T98269 C76ORY 44276517 Ki = 7200 nM T98269 C3AM9S 44276518 Ki = 2200 nM T98269 CRG50V 44276520 Ki = 40 nM T98269 CXP9F3 44276529 Ki = 530 nM T98269 CT6JI8 44276540 Ki = 0.15 nM T98269 C4SMG5 44276541 Ki = 0.2 nM T98269 CY67TF 44276575 Ki = 10 nM T98269 CY7N6P 44276576 Ki = 66 nM T98269 C98FNA 44276588 Ki = 7.1 nM T98269 C3JW2Z 44276590 Ki = 25 nM T98269 CAQ7K8 44276591 Ki = 40 nM T98269 CWPQ79 44276592 Ki = 46 nM T98269 C0UB1W 44276605 Ki = 5.3 nM T98269 CJ4N1A 44276606 Ki = 21 nM T98269 C2J6FL 44276631 Ki = 0.15 nM T98269 CQ2E3T 44276632 Ki = 39 nM T98269 CK4W2X 44276670 Ki = 1.8 nM T98269 CJ9TC2 44276671 Ki = 1.4 nM T98269 CRGT53 44279608 Ki = 24000 nM T98269 CT6UW3 44279609 Ki = 67000 nM T98269 C2F6RG 44279636 Ki = 68000 nM T98269 C67OEX 44279649 Ki > 100000 nM T98269 CP63FY 44279661 Ki = 74000 nM T98269 CW85ND 44279666 Ki = 90000 nM T98269 CJC7Q6 44279667 Ki = 23000 nM T98269 C37JIV 44279668 Ki = 20000 nM T98269 CT0L5I 44279669 Ki > 100000 nM T98269 C2ZA6O 44279683 Ki > 100000 nM T98269 C07KSW 44279690 Ki = 42 nM T98269 C1SV8L 44279695 Ki > 100000 nM T98269 C81ZPS 44279696 Ki = 70000 nM T98269 CPR1I5 44279743 Ki = 4400 nM T98269 C7DVS3 44279744 Ki = 27000 nM T98269 C79IGX 44279760 Ki = 500 nM T98269 C0H8TA 44279761 Ki = 320 nM T98269 CF1G5W 44279762 Ki > 18000 nM T98269 C04QWX 44279778 Ki = 1200 nM T98269 C5X9LI 44279876 Ki = 3800 nM T98269 C3SVY4 44280008 Ki > 100000 nM T98269 CHF48O 44280009 Ki = 9500 nM T98269 CFZ3N6 44280034 Ki > 22000 nM T98269 CP0ES5 44280035 Ki = 4000 nM T98269 CCY4P9 44280036 Ki = 2000 nM T98269 C6EJK2 44280086 Ki = 90 nM T98269 CG3R0D 44280088 Ki = 2600 nM T98269 C6C0IL 44280089 Ki > 28000 nM T98269 COYV60 44280119 Ki = 620 nM T98269 C5DGZ4 44283428 IC50 = 22.3 nM T98269 C35FHY 44301469 Ki = 6 nM T98269 CK4Y5N 44301677 Ki = 113 nM T98269 CL15BA 44301678 Ki = 11 nM T98269 C0OD2S 44301679 Ki = 4.7 nM T98269 CP1I3V 44301693 Ki = 2.7 nM T98269 C5OGC6 44301730 Ki = 120 nM T98269 C0MH2N 44302083 Ki = 60 nM T98269 CNFH63 44302084 Ki = 27 nM T98269 C14QKJ 44302085 Ki = 100 nM T98269 CD8WB9 44304162 Ki > 50000 nM T98269 CXQL04 44309551 Ki = 54 nM T98269 C4PM7J 44309578 Ki = 970 nM T98269 CW9HZ8 44309579 Ki = 1300 nM T98269 CNFK24 44309651 Ki = 150 nM T98269 CGLW68 44309778 Ki = 1200 nM T98269 CQZ59D 44309864 Ki = 54 nM T98269 CXZ38R 44314079 Ki = 4500 nM T98269 CDH48M 44314105 IC50 = 742 nM T98269 CQ4CL1 44314492 IC50 = 5 nM T98269 C7DM0B 44314515 IC50 = 936 nM T98269 C1RTL9 44314516 IC50 = 7 nM T98269 C7CM3V 44315452 Ki = 7.5 nM T98269 CT63DO 44315614 Ki > 20000 nM T98269 CTMU12 44315615 Ki = 2400 nM T98269 CJ2BT4 44315617 Ki = 120 nM T98269 C36NJW 44315634 Ki = 50000 nM T98269 C7FCD1 44315652 Ki = 59 nM T98269 CA9DJ1 44315663 Ki > 20000 nM T98269 CN0YC9 44315681 Ki = 2100 nM T98269 CGS24W 44315689 Ki = 42 nM T98269 C15MDV 44315706 Ki = 28 nM T98269 CTU13L 44315737 Ki > 20000 nM T98269 C37LID 44315971 Ki = 500 nM T98269 CW2U6D 44316052 Ki > 20000 nM T98269 C8VHW3 44316064 Ki > 20000 nM T98269 C50SIZ 44316084 Ki > 20000 nM T98269 C43IDW 44323704 Ki > 10000 nM T98269 CG57OJ 44323820 Ki = 4000 nM T98269 CO7U5V 44323993 Ki = 6000 nM T98269 C3U5BI 44323994 Ki = 42000 nM T98269 CWR4M7 44324063 Ki = 10000 nM T98269 CQI38W 44324147 Ki > 100000 nM T98269 C7BCI2 44324148 Ki = 610 nM T98269 CA5KT7 44324178 Ki = 100 nM T98269 C9UTL8 44324179 Ki = 3100 nM T98269 CK89PV 44325864 IC50 = 36 nM T98269 CU36WF 44325934 IC50 = 10400 nM T98269 CBFO04 44326730 Ki = 880 nM T98269 CJU73H 44326739 Ki = 290 nM T98269 CSGW40 44326740 Ki = 900 nM T98269 C6PK9O 44326752 Ki = 110 nM T98269 CWM86U 44326788 Ki = 4200 nM T98269 CA1E4F 44326790 Ki = 100 nM T98269 CE4JX7 44326801 Ki = 1000 nM T98269 CTJ0W9 44326802 Ki = 410 nM T98269 C86VZO 44326804 Ki = 490 nM T98269 C0TB6I 44326823 Ki = 430 nM T98269 CF7D3Z 44326828 Ki = 440 nM T98269 C92DKG 44326829 Ki = 3000 nM T98269 C9Y3JF 44326830 Ki = 24000 nM T98269 CB5TI1 44326866 Ki = 1100 nM T98269 C8R2FB 44326895 Ki = 1600 nM T98269 CC2FZ8 44326964 Ki = 620 nM T98269 CQKB34 44326977 Ki = 450 nM T98269 CAB39E 44331552 IC50 = 843 nM T98269 CE0FW4 44331565 IC50 = 141 nM T98269 C8SZN9 44331566 IC50 = 429 nM T98269 CMFW61 44331567 IC50 = 831 nM T98269 CHYL38 44331577 IC50 = 611 nM T98269 C1I9QH 44331578 IC50 = 1800 nM T98269 C4VGZ1 44331579 IC50 = 521 nM T98269 CRZ01H 44331580 IC50 = 1900 nM T98269 CFOR90 44331674 IC50 = 1100 nM T98269 CK7VI8 44331675 IC50 = 636 nM T98269 CH7GS4 44331676 IC50 > 10000 nM T98269 C4FOD3 44331693 IC50 = 9420 nM T98269 CJY5L2 44331739 IC50 = 2570 nM T98269 C8N2GQ 44331740 IC50 = 1810 nM T98269 CW9K4Q 44331815 IC50 = 538 nM T98269 CT76DG 44331816 IC50 = 2510 nM T98269 CC70GF 44331830 IC50 = 43 nM T98269 CNJ19L 44331876 IC50 = 3140 nM T98269 C46IPA 44331879 IC50 = 1740 nM T98269 CP0Y8M 44331898 IC50 = 50 nM T98269 CF3R6W 44331908 IC50 = 7430 nM T98269 C0S8LV 44331910 IC50 = 6.5 nM T98269 CTM5W1 44331914 IC50 = 4860 nM T98269 C0YZ9O 44331915 IC50 = 2550 nM T98269 CPZ7Q2 44331933 IC50 = 3240 nM T98269 C4NK1S 44331942 IC50 = 50 nM T98269 CXKY19 44331943 IC50 = 10000 nM T98269 C3FC8D 44331944 IC50 = 2300 nM T98269 CH1ZF2 44331953 IC50 = 790 nM T98269 C0QJ8V 44331957 IC50 = 250 nM T98269 C1HBX6 44331963 IC50 = 18820 nM T98269 C7UXK5 44331964 IC50 = 5850 nM T98269 C42PGN 44331965 IC50 = 330 nM T98269 C5J7KX 44331966 IC50 > 10000 nM T98269 CG83FS 44331967 IC50 = 13700 nM T98269 CGAJ95 44331977 IC50 = 2960 nM T98269 CCYX84 44331980 IC50 = 336 nM T98269 C5UIO2 44331987 IC50 = 1830 nM T98269 C0PM5C 44332004 IC50 = 1860 nM T98269 C4ENB1 44332005 IC50 = 127 nM T98269 CFK4Z1 44332024 IC50 = 3990 nM T98269 CTM3G2 44332026 IC50 = 563 nM T98269 C48ZEW 44332028 IC50 = 35300 nM T98269 C30MKG 44332029 IC50 = 44200 nM T98269 C7OS9X 44332050 IC50 = 2400 nM T98269 C9Y6NP 44332051 IC50 = 650 nM T98269 C0VGF8 44332058 IC50 = 1430 nM T98269 CQU84D 44332068 IC50 = 2210 nM T98269 CBL91D 44332078 IC50 = 2200 nM T98269 C4VCM3 44332093 IC50 = 1320 nM T98269 C92QVT 44332108 IC50 = 2750 nM T98269 CQLZ09 44332109 IC50 = 6840 nM T98269 C4CUL6 44332112 IC50 = 2180 nM T98269 CN2YM6 44332113 IC50 = 1890 nM T98269 C4CY8K 44332118 IC50 = 15 nM T98269 CXZ2N1 44332120 IC50 = 5140 nM T98269 CD56PK 44332121 IC50 = 5250 nM T98269 C5A6OJ 44332128 IC50 = 1800 nM T98269 C6IZ2R 44332129 IC50 = 792 nM T98269 C5DY0G 44332136 IC50 = 385 nM T98269 CQ1K9H 44332311 IC50 = 33 nM T98269 C9LOS2 44332330 IC50 = 686 nM T98269 C2U6GB 44332331 IC50 = 543 nM T98269 CH01QW 44332332 IC50 = 408 nM T98269 C5CV1J 44338023 Ki = 15 nM T98269 CAK8H9 44341482 Ki = 6300 nM T98269 C0UC7G 44341675 IC50 = 46 nM T98269 C0G3VZ 44341677 IC50 = 0.11 nM T98269 CZ0UB6 44341678 IC50 = 0.37 nM T98269 C3C7GQ 44341685 Ki = 10000 nM T98269 CPG70J 44341704 IC50 = 1.9 nM T98269 CE5MI0 44341705 Ki = 14000 nM T98269 CP34CX 44341715 Ki = 240 nM T98269 C5KO8Z 44341732 IC50 = 10 nM T98269 CJ7U0R 44341744 Ki = 260 nM T98269 CIX62Q 44341753 IC50 = 9 nM T98269 CI50SR 44341760 Ki = 14 nM T98269 CQ26VE 44341819 Ki = 160 nM T98269 C9PV0D 44341820 IC50 = 13 nM T98269 CAWK09 44341825 Ki = 8800 nM T98269 CEHX54 44341826 Ki = 13000 nM T98269 CHK85L 44341856 IC50 = 1.7 nM T98269 C7BCF0 44341863 IC50 = 0.4 nM T98269 CIM3V6 44341895 IC50 = 36 nM T98269 C04XTQ 44341930 IC50 = 38 nM T98269 CY9V2J 44341962 IC50 = 2 nM T98269 C1TXN0 44341963 IC50 = 9 nM T98269 C4IN5B 44341984 IC50 = 17 nM T98269 CP3UN9 44342099 Ki = 5 nM T98269 C0EAY7 44342283 Ki = 0.37 nM T98269 CFA9L4 44342718 Ki = 54 nM T98269 C8D5TB 44364680 Ki = 1500 nM T98269 CX3V9O 44379442 Ki = 4 nM T98269 CW3C5B 44379468 Ki = 134 nM T98269 CJF2V1 44379693 Ki = 119000 nM T98269 CGZ5E8 44379781 Ki = 23.9 nM T98269 CAO6L1 44384790 Ki = 410 nM T98269 CKG30Z 44384791 Ki = 11.25 nM T98269 CNI74D 44384792 Ki = 45 nM T98269 CP63UR 44384817 Ki = 57.5 nM T98269 CP9W8C 44384818 Ki = 1650 nM T98269 CMBV36 44384819 Ki = 395 nM T98269 CL6Y4K 44384857 Ki = 78 nM T98269 CHX40L 44384858 Ki = 58 nM T98269 C78VOK 44384930 Ki = 4.8 nM T98269 C1H4RO 44384931 Ki = 25 nM T98269 C5QX7S 44384984 Ki = 0.76 nM T98269 CQVS19 44385001 Ki = 8 nM T98269 C3Q4SW 44385002 Ki = 11.6 nM T98269 COI9Y1 44385003 Ki = 62.5 nM T98269 CF79UR 44385068 Ki = 2.3 nM T98269 C74LEY 44385069 Ki = 1.79 nM T98269 C4IM9P 44385480 Ki = 1.15 nM T98269 CX65ZB 44385481 Ki = 0.85 nM T98269 C12GKJ 44385526 Ki = 34.3 nM T98269 CCK82G 44385577 Ki = 81 nM T98269 C9J4YB 44385696 Ki = 117 nM T98269 C12KVR 44385703 Ki = 37 nM T98269 CR08QD 44385704 Ki = 2.39 nM T98269 C3VFE8 44385705 Ki = 3.1 nM T98269 CDQT94 44385921 Ki = 3.05 nM T98269 CT2ZL7 44386278 Ki = 22.8 nM T98269 CB85GE 44386279 Ki = 7.3 nM T98269 CZK39M 44386280 Ki = 4 nM T98269 C7KUY4 44386337 Ki = 255 nM T98269 CV23MO 44389236 IC50 = 0.73 nM T98269 C2I3VJ 44389240 IC50 = 0.06 nM T98269 CI89LR 44389245 IC50 = 0.89 nM T98269 CR7VM8 44389295 IC50 = 0.98 nM T98269 CU5VW3 44389297 IC50 = 0.064 nM T98269 C5P8TU 44389299 IC50 = 1.75 nM T98269 C5YC0O 44389306 IC50 = 0.29 nM T98269 C1FMX8 44389307 IC50 = 1.14 nM T98269 CB6US3 44389310 IC50 = 1.7 nM T98269 CC8S0I 44389315 IC50 = 0.22 nM T98269 CEO19T 44389316 IC50 = 0.056 nM T98269 CRC82Z 44389318 IC50 = 1.9 nM T98269 CPE0S2 44389319 IC50 = 0.62 nM T98269 CC8MG3 44389324 IC50 = 1.6 nM T98269 C9X1RJ 44389325 IC50 = 0.15 nM T98269 CF0CN3 44389326 IC50 = 0.62 nM T98269 C7LQP0 44389331 IC50 = 0.88 nM T98269 CEQ2L1 44389335 IC50 = 1.11 nM T98269 C9C3JB 44389337 IC50 = 0.031 nM T98269 CU0I3N 44389338 IC50 = 0.013 nM T98269 CALT41 44389340 IC50 = 1.23 nM T98269 C5LO3T 44389347 IC50 = 0.0087 nM T98269 CJA5K7 44389348 IC50 = 0.047 nM T98269 C2WS9G 44389351 IC50 = 5.13 nM T98269 CEH8Z5 44389369 IC50 = 0.028 nM T98269 CBJ15U 44389458 IC50 = 0.048 nM T98269 C2OU7Z 44389483 IC50 = 0.025 nM T98269 CA81WI 44389513 IC50 = 0.025 nM T98269 CL4G2Y 44389531 IC50 = 0.063 nM T98269 CX5Y3A 44389532 IC50 = 0.067 nM T98269 CEH02Q 44389544 IC50 = 0.11 nM T98269 CXN03I 44389545 IC50 = 0.11 nM T98269 CQPY50 44391346 IC50 = 6505 nM T98269 CJQE23 44391364 IC50 > 10000 nM T98269 CE3YN5 44391369 IC50 > 10000 nM T98269 CWVF04 44391384 IC50 > 10000 nM T98269 C0J6SU 44391388 IC50 = 5810 nM T98269 C24KOF 44391455 IC50 > 10000 nM T98269 CA58XR 44391530 IC50 = 4490 nM T98269 CU3ZB5 44391569 IC50 = 1540 nM T98269 CI7F3G 44391602 IC50 = 4850 nM T98269 CL73OE 44391603 IC50 = 2460 nM T98269 CIU0P1 44391632 IC50 = 675 nM T98269 C5J4LV 44403257 IC50 = 44 nM T98269 CYNX83 44403316 IC50 = 30 nM T98269 CAGR97 44403319 IC50 = 38 nM T98269 CWQ21I 44403320 IC50 15 nM T98269 C5P9KT 44403321 IC50 22 nM T98269 CB2E3T 44403325 IC50 24 nM T98269 CAU6G0 44404870 IC50 = 55 nM T98269 CU4N7M 44404871 IC50 = 97 nM T98269 C3RL0N 44404877 IC50 = 421 nM T98269 CGQ1U4 44404931 IC50 = 4583 nM T98269 CKU1S0 44404937 IC50 = 264 nM T98269 CO38AJ 44405528 IC50 = 10 nM T98269 CBY58A 44405529 IC50 = 5 nM T98269 CVJ8Z3 44405532 IC50 = 6 nM T98269 CHG69W 44405540 IC50 = 1 nM T98269 CZ8Y2S 44405566 IC50 = 1 nM T98269 C6X1JT 44405629 IC50 = 1 nM T98269 CK62FC 44405634 IC50 = 1 nM T98269 COXU97 44405637 IC50 = 1 nM T98269 CGV2B4 44405663 IC50 = 1 nM T98269 CFX81S 44405672 IC50 = 7 nM T98269 CS40LN 44405689 IC50 = 1 nM T98269 C2MOF9 44405695 IC50 = 1 nM T98269 CYG86L 44405707 IC50 = 6 nM T98269 CMUS37 44405733 IC50 = 2 nM T98269 CJ07FL 44405737 IC50 = 5 nM T98269 C1VY3T 44405740 IC50 = 1 nM T98269 C0DL8M 44405752 IC50 = 1 nM T98269 CB7V6W 44405784 IC50 = 3 nM T98269 C1VW8E 44405799 IC50 = 74 nM T98269 CH6CN5 44405800 IC50 = 50 nM T98269 C8EK9W 44405805 IC50 = 9 nM T98269 CWP51F 44405816 IC50 = 135 nM T98269 CEY48X 44405818 IC50 = 130 nM T98269 CXA87L 44405820 IC50 = 3 nM T98269 CM2GJ1 44405827 IC50 = 33 nM T98269 CAY57C 44405829 IC50 = 7 nM T98269 C7LEI3 44405837 IC50 = 3 nM T98269 CFZQ05 44407017 Ki = 1000 nM T98269 CF4CO7 44407019 Ki = 4 nM T98269 C4E8WT 44407042 Ki = 2100 nM T98269 CY7FI8 44407051 Ki = 7 nM T98269 CK2E0R 44407052 Ki = 37000 nM T98269 C53UXL 44407053 Ki = 100 nM T98269 CD3P5X 44407056 Ki = 16 nM T98269 CBD6O5 44407057 Ki = 120 nM T98269 C9CK0X 44407060 Ki = 5 nM T98269 CP1F3H 44407067 Ki = 5 nM T98269 CD8GZ0 44407077 Ki = 8 nM T98269 CDL39P 44407097 Ki = 320 nM T98269 C0G9SW 44407102 Ki = 4 nM T98269 C3OX5B 44407108 Ki = 54 nM T98269 CBP7T6 44407110 Ki = 100 nM T98269 C0DVW2 44407111 Ki = 2100 nM T98269 COYW01 44407122 Ki = 5200 nM T98269 C5OFP7 44407123 Ki = 2800 nM T98269 C6JY9U 44407128 Ki = 1950 nM T98269 CGCN74 44407132 Ki = 35 nM T98269 CF7R0B 44407139 Ki = 2400 nM T98269 C45ENI 44407143 Ki = 43 nM T98269 CS30ZJ 44407152 Ki = 2600 nM T98269 CB9PR2 44407157 Ki = 260 nM T98269 CUY3M1 44414212 IC50 = 30 nM T98269 C79OFE 44414311 IC50 = 2900 nM T98269 CFL7O1 44414418 IC50 = 580 nM T98269 C2DIQ3 44414439 IC50 = 50 nM T98269 C9Q4KR 44414440 IC50 = 240 nM T98269 C0FQ1E 44414442 IC50 = 430 nM T98269 C50NAG 44414456 IC50 = 200 nM T98269 C34DMY 44414457 IC50 = 490 nM T98269 CV0EW7 44414458 IC50 = 50 nM T98269 CL29BC 44414459 IC50 = 90 nM T98269 CV96AO 44414484 IC50 >= 10000 nM T98269 C9P7ZA 44414485 IC50 = 700 nM T98269 C4GWP5 44414501 IC50 = 430 nM T98269 CY0VU1 44414502 IC50 = 40 nM T98269 C8H5YL 44414541 IC50 = 260 nM T98269 CW45EL 44414543 IC50 = 40 nM T98269 CB0M5Q 44414572 IC50 = 310 nM T98269 CXEH76 44414573 IC50 = 150 nM T98269 CMI4Z9 44414574 IC50 = 240 nM T98269 CJT30G 44414592 IC50 = 150 nM T98269 CIQ36K 44414642 IC50 >= 10000 nM T98269 CW0MH5 44416221 IC50 = 2300 nM T98269 COS6D2 44416249 IC50 = 320 nM T98269 CL6YM3 44416250 IC50 = 130 nM T98269 CL8IC5 44416262 IC50 = 150 nM T98269 C21FST 44416320 IC50 = 350 nM T98269 C3FO6V 44416321 IC50 = 150 nM T98269 CN91HB 44416330 IC50 = 80 nM T98269 CF6J2T 44416331 IC50 = 70 nM T98269 CJ6QG4 44417479 IC50 > 60000 nM T98269 C7RX9I 44418960 Ki = 6.3 nM T98269 C4A3MT 44428499 IC50 = 4 nM T98269 C9EIP7 44428502 IC50 = 3 nM T98269 C9E5QZ 44428504 IC50 = 77 nM T98269 C0YBP2 44428506 IC50 = 27 nM T98269 CY3K9C 44428508 IC50 = 14 nM T98269 CF2NM3 44428511 IC50 = 20 nM T98269 CD9VU2 44428513 IC50 = 168 nM T98269 CT8R6X 44428515 IC50 = 53 nM T98269 CS87UF 44428517 IC50 = 11 nM T98269 C12AHI 44428519 IC50 = 29 nM T98269 CWG6S2 44428521 IC50 = 15 nM T98269 CYHS50 44428523 IC50 = 1 nM T98269 CERS10 44428524 IC50 = 13 nM T98269 C2Q0FD 44428525 IC50 = 19 nM T98269 C9R5MT 44428526 IC50 = 22 nM T98269 C3CY9O 44428527 IC50 = 8 nM T98269 CM50ES 44428528 IC50 = 7 nM T98269 CP3XJ0 44428530 IC50 = 3 nM T98269 C62JNP 44428532 IC50 = 2 nM T98269 C5AE0W 44428534 IC50 = 2 nM T98269 CE0V2J 44428536 IC50 = 1 nM T98269 CL6K0W 44428539 IC50 = 1 nM T98269 CXR1V5 44434249 IC50 = 12 nM T98269 C31JIN 44438441 IC50 = 5490 nM T98269 CKI30F 44438442 IC50 = 2310 nM T98269 CNO1C0 44438443 IC50 = 320 nM T98269 CI1G7O 44438444 IC50 = 330 nM T98269 C7GF9S 44577362 IC50 = 330 nM T98269 C48UCA 45379520 Ki = 600 nM T98269 C5Y1IC 45379628 Ki = 47 nM T98269 C15GRV 45379629 Ki = 1200 nM T98269 C8Y9PV 45379630 Ki = 965 nM T98269 CB5NR3 45379631 Ki = 1370 nM T98269 CW25LU 45379632 Ki = 1820 nM T98269 C7ILQ6 45379730 Ki = 209 nM T98269 CD49WC 45379731 Ki = 945 nM T98269 CL39XB 45379732 Ki = 1890 nM T98269 CIFZ76 45379733 Ki = 128 nM T98269 C48VCS 45379836 Ki > 50000 nM T98269 CNH47R 45379837 IC50 = 0.2 nM T98269 C4OW3A 46933234 Ki = 15000 nM T98269 C3OTU4 46933235 Ki = 7 nM T98269 CZ57BW 46934568 Ki = 500 nM T98269 CDY2W5 49796910 IC50 = 0.05 nM T98269 C0HMT1 49797331 IC50 = 3.4 nM T98269 CFZ53P 49864317 Ki = 115 nM T98269 CQ75LB 49864318 Ki = 70.9 nM T98269 CDI0Y3 49864337 Ki = 118 nM T98269 C3G2UJ 49864338 Ki = 16.9 nM T98269 CWZ41D 49864339 Ki = 100 nM T98269 CH1S9N 49864340 Ki = 9.24 nM T98269 CP3LA2 49864341 Ki = 21.5 nM T98269 C1I6AW 49864361 Ki = 0.95 nM T98269 CLC2H0 49864362 Ki = 1020 nM T98269 COGK30 49864363 Ki = 0.58 nM T98269 C7UW4B 49864364 Ki = 5.02 nM T98269 CS43NW 49864365 Ki = 7.9 nM T98269 CXH72O 49864383 Ki = 1.29 nM T98269 CUA2J0 49864384 Ki = 0.9 nM T98269 C4OA6Y 49864385 Ki = 4.03 nM T98269 CSK34F 49864386 Ki = 20 nM T98269 CF7B6N 49864387 Ki = 4.85 nM T98269 C6O8LR 49864398 Ki = 2.81 nM T98269 C6UJ8T 49864399 Ki = 4.68 nM T98269 C6KW0J 49864400 Ki = 3.85 nM T98269 CM86HZ 49864401 Ki = 1.26 nM T98269 CV12MO 49864418 Ki = 1.31 nM T98269 CQ52WY 49864419 Ki = 3 nM T98269 CLQ25K 49864420 Ki = 1.81 nM T98269 CY7J4W 49864421 Ki = 16.7 nM T98269 CWV1I9 49864448 Ki = 4.3 nM T98269 C0FOM2 49864837 Ki = 119000 nM T98269 C8NE0J 49864838 Ki = 8300 nM T98269 CRZO97 49864881 Ki = 16000 nM T98269 CY18LI 49864882 Ki = 1700 nM T98269 C1NHT0 49864883 Ki = 1100 nM T98269 C7X1EG 49864884 Ki = 5600 nM T98269 CG62QR 49864922 Ki = 6000 nM T98269 CIMF98 49864923 Ki = 1300 nM T98269 CM8E0R 49864924 Ki = 1000 nM T98269 C3CPI5 49864963 Ki = 1000 nM T98269 C1AN7G 49864964 Ki = 4400 nM T98269 CC64QE 49864965 Ki = 1300 nM T98269 CXH6A1 49864966 Ki = 2000 nM T98269 CI2MW1 49865022 Ki = 8500 nM T98269 C5N7EK 49865023 Ki = 800 nM T98269 C6YI9H 49865024 Ki = 1100 nM T98269 C30SUT 49865025 Ki = 600 nM T98269 CJ0HK1 49865079 Ki = 800 nM T98269 C5V0IL 49865080 Ki = 1200 nM T98269 CO1KM9 49865081 Ki = 2600 nM T98269 CEPK96 49865138 Ki = 87200 nM T98269 CRPL58 49865139 Ki = 9200 nM T98269 CIN12P 49865140 Ki = 17500 nM T98269 COL0H6 49865193 Ki = 14000 nM T98269 CO2V3K 49865194 Ki = 21000 nM T98269 CVIQ74 49865195 Ki = 66500 nM T98269 CXIO14 49865196 Ki = 27500 nM T98269 C90UWA 49865247 Ki = 84000 nM T98269 C43IYW 49865248 Ki = 298000 nM T98269 C2M4OT 49865249 Ki = 1500 nM T98269 CDA8T3 49865250 Ki = 134 nM T98269 C9H7QU 49865251 IC50 = 2 nM T98269 C2M0PB 49865252 Ki = 1 nM T98269 CGQ1O0 49865253 Ki = 2 nM T98269 C63FWH 49865255 Ki = 1 nM T98269 CN8L7W 51723030 IC50 = 90000 nM T98269 C3M2BW 52918163 IC50 > 10000 nM T98269 CF24IM 52918177 IC50 > 20000 nM T98269 CR9I7F 52918178 IC50 > 20000 nM T98269 C2VPU1 52918179 IC50 > 20000 nM T98269 C8Z2TQ 54580470 IC50 > 50000 nM T98269 CMU0B4 54581481 IC50 > 25000 nM T98269 CCS8Y3 54581987 IC50 > 10000 nM T98269 CJEP38 54582484 IC50 > 50000 nM T98269 C61NWL 54582924 IC50 > 50000 nM T98269 CO0AG3 54583923 IC50 = 4775 nM T98269 CI2DL4 54583924 IC50 > 50000 nM T98269 CV2WU1 54583925 IC50 > 20000 nM T98269 CXA51D 54584867 IC50 > 20000 nM T98269 C8YSL0 54585834 IC50 = 5733 nM T98269 C9B5OF 54586343 IC50 > 25000 nM T98269 C7A8ER 54587376 IC50 > 15000 nM T98269 C5O9SR 57333875 IC50 = 100000 nM T98269 CGY3W2 71471109 IC50 = 1050 nM T98269 CKZ2H0 71582971 IC50 = 12100 nM T98269 C4WJ5F 71582972 IC50 = 15500 nM T98269 CXA62J 71582973 IC50 = 7340 nM T98269 CNZS31 71582974 IC50 = 11600 nM T98269 CE4L9D 71582975 IC50 > 500000 nM T98269 CXMS80 71583078 IC50 > 500000 nM T98269 C30UIL 71583079 IC50 > 500000 nM T98269 CJBC14 71583080 IC50 = 18400 nM T98269 C57MOP 71583081 IC50 > 500000 nM T98269 CS0YK9 71583082 IC50 = 18400 nM T98269 C3UTO9 71583083 IC50 = 24700 nM T98269 CW1R5Q 71583084 IC50 = 45800 nM T98269 CR57LS 71583192 IC50 = 14700 nM T98269 C8B3NZ 71583193 IC50 = 25900 nM T98269 CB6DY7 71583194 IC50 = 30700 nM T98269 CANH70 71716242 IC50 = 13200 nM T98269 C40WIR 71718085 IC50 = 26 nM T98269 CU75VK 71719897 IC50 = 2700 nM T98269 CBV6F1 71720507 IC50 = 20 nM T98269 C1QX3B 73345613 Ki = 1.1 nM T98269 C4U5TO 76311196 IC50 = 4695 nM T98269 CSI53E 76311200 IC50 > 10000 nM T98269 CNOL37 76311201 IC50 = 522 nM T98269 C8IS5Q 76314800 IC50 = 672 nM T98269 CK41QI 76314804 IC50 = 1697 nM T98269 CHS61N 76314805 IC50 > 10000 nM T98269 CDY7K0 76318413 IC50 > 10000 nM T98269 CB2N6G 76322078 IC50 > 10000 nM T98269 C8SPW6 76322082 IC50 > 10000 nM T98269 CC2EP6 76325698 IC50 > 10000 nM T98269 CFY79U 76332916 IC50 > 10000 nM T98269 CD35SI 76332917 IC50 = 1878 nM T98269 C3FQX0 76336535 IC50 > 10000 nM T98269 CV4PE6 76336536 IC50 > 10000 nM T98269 CKCI60 90663142 IC50 = 87 nM T98269 C9BL3E 90663191 IC50 = 1 nM T98269 CYW35T 90663634 Ki = 4900 nM T98269 CF83WN 90663635 Ki = 1700 nM T98269 C3GPO7 118723314 IC50 = 500000 nM T98269 C8H0EL 118723315 IC50 = 500000 nM T98269 CTE1O2 118723316 IC50 = 500000 nM T98269 CE8O9P 118723317 IC50 = 500000 nM T98269 C48DEF 118723325 IC50 = 500000 nM T98269 C67QMY 118723326 IC50 = 500000 nM T98269 CCJ27M 118723327 IC50 = 500000 nM T98269 COG92V 118723328 IC50 = 2590 nM T98269 CSX85P 118723329 IC50 = 500000 nM T98269 CICB42 118723330 IC50 = 9970 nM T98269 C13BRQ 118723331 IC50 = 7430 nM T98269 C52FZR 127028674 IC50 = 150000 nM T98269 CR19OH 127028675 IC50 = 25000 nM T98269 C8KE7R 127028996 IC50 = 50000 nM T98269 CWM2E8 133081971 IC50 = 9.8 nM T98269 CID3N6 134134572 Ki = 202 nM T98269 CV0R3B 134135432 Ki = 227 nM T98269 C3D7LQ 134136688 Ki = 534 nM T98269 CBY95D 134138690 Ki = 200 nM T98269 CG3EI1 134145896 Ki = 49 nM T98269 CI9X3K 134147411 Ki = 16 nM T98269 CP16IA 134148745 Ki = 75 nM T98269 CPE90G 134149983 Ki = 303 nM T98269 CBE39C 134151245 Ki = 183 nM T98269 CY0LD4 134152014 Ki = 27 nM T98269 C3K5HR 134153309 Ki = 59 nM T98269 CWQT79 134156687 Ki = 129 nM T98269 CJ3B6S 145708113 IC50 = 86 nM T98269 CZ70SI 145963799 IC50 > 10000 nM T98269 COE9X7 145964860 IC50 = 5011.87 nM T98269 CYCR59 145965957 IC50 = 66 nM T98269 CIFO51 145966058 IC50 = 31.62 nM T98269 CJTQ64 145966473 IC50 = 23 nM T98269 CI4F7K 145967000 IC50 > 10000 nM T98269 CZ3F6G 145967287 IC50 = 1258.93 nM T98269 CMH8B6 145968964 IC50 = 501.19 nM T98269 CD8EL9 145972318 IC50 > 10000 nM T98269 CHJS10 145972560 IC50 = 21 nM T98269 CJE42P 145972735 IC50 > 10000 nM T98269 CM92VF 145973492 IC50 = 4.7 nM T98269 C83TKO 145973689 IC50 > 10000 nM T98269 CP4KZ5 145974701 IC50 = 360 nM T98269 C9CI3O 145975395 IC50 = 11 nM T98269 CY07KF 145975559 IC50 = 53 nM T98269 C5QJ7R 145975761 IC50 > 10000 nM T98269 C1HC2G 145976171 IC50 = 76 nM T98269 C6FU3Q 145976723 IC50 = 39.81 nM T98269 CSZ92C 145977507 IC50 = 200 nM T98269 CCQ51X 145977563 IC50 = 15.85 nM T98269 CDL16P 145978002 IC50 = 50 nM T98269 CF6U1Q 145978382 IC50 = 210 nM T98269 CR2S0C 108068 Ki = 10600 nM T98269 D0L9AX 644345 IC50 = 190 nM T98269 D0M2EM 4650 IC50 = 3000 nM T98269 D0N5MU 4117381 Ki = 9000 nM T98269 D0P3XJ 44407073 Ki = 180 nM T98269 D0Q9XX 515950 Ki = 12000 nM T98269 D0X8XO 10112904 Ki = 8 nM T98269 D0Y5IQ 44255320 IC50 = 5000 nM T98539 C08KEM 122179540 IC50 = 5500 nM T98539 C3AJ4C 122179546 IC50 = 6500 nM T98539 CG0RP7 122179547 IC50 = 4300 nM T98539 C1A0SQ 122179548 IC50 = 5500 nM T61722 D0R1RS 3715 Ki = 50 nM T61722 D0WL5V 9867642 Ki = 745 nM T61722 D0YB1G 28871 IC50 = 550 nM T61722 D0GC5H 123879 Ki = 4.3 nM T61722 D0I3TU 45268455 IC50 = 2.2 nM T61722 D0K1EG 11508736 IC50 = 3 nM T61722 D0RL4X 45270144 IC50 = 42 nM T61722 D0SP5V 49843471 IC50 = 30 nM T61722 D0T4SG 11292191 IC50 = 4.3 nM T61722 D0U1HN 44158492 IC50 = 4.9 nM T61722 D0X7EG 11462174 Ki = 13 nM T61722 D0YB2Y 42641863 IC50 = 3 nM T61722 CYFR68 5036 Ki = 5.5 nM T61722 C3W5UX 7204 Ki > 10000 nM T61722 CF9B2G 184853 IC50 = 1300 nM T61722 CO9ZR3 198256 IC50 > 100000 nM T61722 CB9I8Y 262282 IC50 = 158 nM T61722 CC21JK 570211 IC50 > 50000 nM T61722 CVGZ96 626746 IC50 = 794 nM T61722 CYCJ10 797803 IC50 = 430 nM T61722 CG4XM1 810847 IC50 = 388 nM T61722 CAMZ27 810849 IC50 = 881 nM T61722 CW01HG 950344 IC50 = 350 nM T61722 CYP6M5 1001787 IC50 = 210 nM T61722 CFG9T5 1101166 EC50 = 11 nM T61722 CNZ0G7 1101168 IC50 > 10000 nM T61722 CE84TM 1101169 IC50 = 420 nM T61722 CN4A5M 1208785 IC50 = 450 nM T61722 CQ29PI 1268975 IC50 = 500 nM T61722 CT53UG 1282226 IC50 = 1300 nM T61722 C2UQ7Y 2178182 IC50 = 84 nM T61722 C7CYB4 2763924 IC50 = 990 nM T61722 CYE1K0 2772433 IC50 = 2370 nM T61722 C61AVS 2772705 IC50 = 590 nM T61722 CLU85B 2772717 IC50 = 2500 nM T61722 C5GI9F 2772718 IC50 = 2000 nM T61722 C6VQU0 2835229 IC50 = 34 nM T61722 CSC0J3 2837129 IC50 > 50000 nM T61722 CO7HE3 2848830 IC50 = 6600 nM T61722 C3NW1B 3054243 IC50 = 440 nM T61722 CPW8B3 3091947 IC50 = 64 nM T61722 CNIH29 3135989 IC50 = 9 nM T61722 C78GEV 3145335 IC50 = 130 nM T61722 C4S8GO 3145349 IC50 = 49 nM T61722 CQR7M9 3145355 IC50 = 89 nM T61722 CCS63D 3145374 IC50 = 96 nM T61722 CL0EK8 3145377 IC50 = 960 nM T61722 C69VBT 3159627 IC50 = 5500 nM T61722 CY4FN7 3479396 IC50 = 1460 nM T61722 CMT5I6 3568495 IC50 = 990 nM T61722 C0PBW1 3753058 IC50 = 105 nM T61722 CFR95D 3880137 IC50 = 1400 nM T61722 CBL68W 4033797 IC50 = 1300 nM T61722 C74JYQ 4100224 IC50 = 940 nM T61722 CTG1A2 4151295 IC50 = 390 nM T61722 CDG6K5 4151297 IC50 = 350 nM T61722 CEC52U 4151299 IC50 = 460 nM T61722 CRPS18 4151301 IC50 = 4100 nM T61722 C9QW2U 4151303 IC50 = 210 nM T61722 CI2NF6 4261307 IC50 = 7000 nM T61722 CE7LS5 5197257 IC50 = 3620 nM T61722 C2XZ4K 5290618 IC50 = 210 nM T61722 CYNX02 5333629 IC50 = 555 nM T61722 C4Z7XU 5344298 IC50 = 11200 nM T61722 CJ8P4T 5352624 Ki = 3500 nM T61722 C24HIW 5722969 IC50 = 3660 nM T61722 CLV80X 5726103 IC50 = 12800 nM T61722 CM4AB0 6461002 Ki > 10000 nM T61722 CY36TK 6519333 EC50 = 7 nM T61722 C26SZF 7097677 IC50 = 180 nM T61722 CB5DJ4 7097680 IC50 = 15 nM T61722 CQA35F 9802748 Ki = 1.9 nM T61722 CXI27J 9872340 IC50 = 3 nM T61722 C7Y1MF 9884103 IC50 = 79 nM T61722 CKIE37 9985715 IC50 = 2 nM T61722 C0KIT3 9999681 IC50 = 79 nM T61722 CZ39MP 10020475 IC50 = 15 nM T61722 CR7QC1 10021510 IC50 = 1000 nM T61722 C3FKC4 10021783 IC50 = 25 nM T61722 C2BF4G 10022229 IC50 = 71 nM T61722 C45TBJ 10023245 IC50 = 1.4 nM T61722 C9VX0B 10042953 IC50 = 7.1 nM T61722 CAE21W 10043211 IC50 = 2.6 nM T61722 CVB57E 10046404 IC50 = 6 nM T61722 CUW28C 10047003 IC50 = 3.5 nM T61722 CLA97I 10047141 IC50 = 71 nM T61722 CPOJ20 10047280 IC50 = 126 nM T61722 CN1H0Q 10065219 IC50 = 21 nM T61722 C7HQ6R 10066327 IC50 = 7.1 nM T61722 C81RJV 10069458 IC50 = 1750 nM T61722 CIKF91 10069991 IC50 = 1 nM T61722 C4TL3V 10090208 IC50 = 2.3 nM T61722 CQP3F8 10090285 IC50 = 42 nM T61722 C15PXG 10095612 IC50 = 7.9 nM T61722 C6NT2P 10098978 IC50 = 4 nM T61722 C1KF3U 10237369 IC50 = 180 nM T61722 C6PMT7 10249850 IC50 = 178 nM T61722 CP1I7X 10251489 IC50 = 93 nM T61722 CGXU05 10316809 IC50 = 60 nM T61722 CBH29S 10317477 IC50 = 178 nM T61722 C7AY2L 10337564 IC50 = 2.6 nM T61722 C0A6IO 10340798 IC50 = 5.4 nM T61722 CHG82R 10384259 IC50 = 13 nM T61722 C9W0UP 10405318 IC50 = 3 nM T61722 CSO29N 10407275 IC50 = 26 nM T61722 C3NS9H 10407503 IC50 = 7.1 nM T61722 CEO91X 10409908 IC50 = 7.1 nM T61722 CLD09V 10428273 IC50 = 18 nM T61722 CXK1N4 10430988 IC50 = 430 nM T61722 CZ0I6Y 10473927 IC50 = 1.3 nM T61722 CZ1XW6 10483360 Ki = 1 nM T61722 CFS2N7 11154496 IC50 = 1.8 nM T61722 C3PE6A 11175439 Ki = 15 nM T61722 CV70CO 11176300 Ki = 7 nM T61722 CR36QL 11187351 Ki = 6 nM T61722 CU06DP 11189402 IC50 = 293 nM T61722 CZJU57 11195860 IC50 = 708 nM T61722 CQL79W 11222822 IC50 = 11 nM T61722 CNU4B3 11245359 Ki = 457 nM T61722 CJ87PV 11258980 IC50 = 1.3 nM T61722 C4KG3Y 11281300 IC50 = 0.6 nM T61722 C92FAZ 11301859 Ki = 634 nM T61722 CNT89F 11315250 IC50 = 56 nM T61722 C30EIV 11325699 IC50 = 19 nM T61722 C0KN2O 11326126 IC50 = 4.1 nM T61722 CWH1S9 11336492 IC50 = 50 nM T61722 C10OIJ 11360614 IC50 = 32 nM T61722 C32ZCI 11382433 Ki = 9 nM T61722 CB0N6G 11382710 IC50 = 8.9 nM T61722 CFK86C 11403482 IC50 = 10 nM T61722 C7DLM6 11405875 IC50 = 8 nM T61722 CVWY92 11407412 IC50 = 224 nM T61722 CK7D1E 11407637 Ki = 68 nM T61722 C7IOQ3 11416126 IC50 = 251 nM T61722 C6QLE7 11452761 IC50 = 9.7 nM T61722 CZ4K0P 11476788 Ki = 19200 nM T61722 CX74JM 11482181 IC50 = 251 nM T61722 CORM68 11485353 Ki = 2979 nM T61722 CHG40L 11494022 Ki = 109 nM T61722 CH4G7C 11494161 IC50 = 15 nM T61722 C4QUK1 11494321 Ki = 225 nM T61722 CIC10G 11494396 IC50 = 820 nM T61722 CI4PY3 11494496 IC50 = 8 nM T61722 CW3YO5 11494768 IC50 = 40 nM T61722 CG4I5C 11495505 IC50 = 36 nM T61722 CZQO56 11495838 IC50 = 14 nM T61722 C0F8HO 11496258 IC50 = 3.5 nM T61722 CY1XS8 11500800 IC50 = 475 nM T61722 CQ6IU7 11509269 IC50 = 14 nM T61722 CL12DX 11511330 IC50 = 12 nM T61722 CWX9U7 11516114 Ki = 377 nM T61722 CD30WO 11516319 Ki = 48 nM T61722 CS2LR0 11516353 IC50 = 42 nM T61722 CB18VF 11517351 IC50 = 14 nM T61722 CJQ60P 11517780 IC50 = 18 nM T61722 CV02QY 11518211 IC50 = 517 nM T61722 CW91TC 11521904 IC50 = 1600 nM T61722 C15UCV 11523333 IC50 = 15 nM T61722 C8L0KR 11530248 IC50 = 51 nM T61722 CX9PN6 11531874 IC50 = 4.1 nM T61722 C4D3UZ 11532160 IC50 = 330 nM T61722 CM7H8E 11532165 IC50 = 30 nM T61722 C39PBD 11536944 Ki = 624 nM T61722 C12FMI 11537570 IC50 = 430 nM T61722 C9FQW8 11537884 Ki = 71 nM T61722 CR6M4N 11539052 IC50 = 316 nM T61722 CF2OM8 11539410 IC50 = 7 nM T61722 CIC1L3 11539725 IC50 = 31 nM T61722 CFW89P 11544651 IC50 = 230 nM T61722 C2B8HY 11545850 Ki = 0.51 nM T61722 C6A3KV 11546947 IC50 = 79 nM T61722 CI8VO0 11547484 IC50 = 1.4 nM T61722 CM7HK0 11551847 IC50 = 70 nM T61722 C7ATR5 11551917 Ki = 619 nM T61722 CP5Z2K 11554216 IC50 = 5.6 nM T61722 C78ZRI 11559328 IC50 = 107 nM T61722 C78FTM 11561470 IC50 = 8.4 nM T61722 C0I8VR 11568356 IC50 = 7.5 nM T61722 CSJP24 11568443 IC50 = 10 nM T61722 CN1O9M 11573030 Ki = 20 nM T61722 C1J4ST 11573244 IC50 = 23 nM T61722 CBCJ63 11573475 Ki = 282 nM T61722 CCWG81 11573514 Ki = 143 nM T61722 CXQD46 11573799 Ki = 250 nM T61722 CE1X0N 11574056 Ki = 2619 nM T61722 C10XRF 11574877 IC50 = 2.5 nM T61722 CI9ED3 11575484 IC50 = 4 nM T61722 CPM6D7 11582965 IC50 = 3 nM T61722 CH0Y3G 11583024 IC50 = 3.5 nM T61722 CM7S6Q 11588648 Ki = 103 nM T61722 C7N9PZ 11590255 IC50 = 631 nM T61722 CCZ7L9 11590561 IC50 = 45 nM T61722 C96TKX 11595451 IC50 = 11 nM T61722 CAZ31O 11597936 IC50 = 1.3 nM T61722 C6KEF0 11603173 IC50 = 4 nM T61722 CE9ZJ0 11604412 IC50 = 71 nM T61722 CJ1RC8 11605389 Ki = 38 nM T61722 CU56NL 11608862 Ki = 588 nM T61722 C8W0FS 11610095 IC50 = 450 nM T61722 C2M8HZ 11610353 IC50 = 30 nM T61722 CQ5WH9 11611100 IC50 = 8.7 nM T61722 CE61GR 11611101 IC50 = 2.9 nM T61722 C8W7JO 11611215 IC50 = 3.5 nM T61722 C50DOT 11618107 IC50 = 80 nM T61722 CJ5R4H 11618108 IC50 = 1.7 nM T61722 CSP67N 11619293 IC50 = 10 nM T61722 C4G7DE 11624420 IC50 = 200 nM T61722 CORL03 11625836 Ki = 19 nM T61722 C0C1SP 11626318 IC50 = 10 nM T61722 C9L5VD 11631813 IC50 = 34 nM T61722 CD7R5P 11631965 IC50 = 62 nM T61722 CK7IJ5 11633473 IC50 = 9 nM T61722 C7PN8S 11633547 IC50 = 1.4 nM T61722 CB31VQ 11633804 IC50 = 6.8 nM T61722 CTV9A4 11639997 IC50 = 71 nM T61722 C72OQN 11640178 IC50 = 1 nM T61722 C7N4ZG 11640298 IC50 = 3.3 nM T61722 C3SFA1 11645962 Ki = 145 nM T61722 CHOG21 11646330 Ki = 106 nM T61722 CTKB78 11646408 IC50 = 60 nM T61722 C5LI7P 11647012 IC50 = 1.5 nM T61722 CQP48G 11648347 IC50 = 3.9 nM T61722 C28FMW 11652270 Ki = 302 nM T61722 CMB6F9 11653874 IC50 = 9 nM T61722 CODZ91 11655069 IC50 = 4.5 nM T61722 C1BXN6 11660316 IC50 = 1010 nM T61722 C6VW9O 11662033 IC50 = 45 nM T61722 CJ4P0D 11667039 Ki = 99 nM T61722 C51UDK 11667741 IC50 = 17 nM T61722 CBSL25 11669738 IC50 = 11 nM T61722 CIUJ01 11670392 IC50 = 4 nM T61722 CWS82F 11673910 Ki = 379 nM T61722 CSE86V 11674088 Ki = 278 nM T61722 CK1W5R 11675066 IC50 = 5 nM T61722 C97FRY 11675335 IC50 = 26 nM T61722 C9Q3ED 11675688 Ki = 52 nM T61722 CXZ9B5 11676516 IC50 = 28 nM T61722 C5PMH6 11681442 IC50 = 210 nM T61722 C5YV7X 11682247 IC50 = 18 nM T61722 C72BNQ 11682521 IC50 = 5 nM T61722 COXZ65 11682932 IC50 = 28 nM T61722 C46KHX 11683632 IC50 = 4 nM T61722 C6NQK1 11688573 IC50 = 5 nM T61722 C0OWD4 11689128 Ki = 3220 nM T61722 CW8RY9 11689895 IC50 = 1 nM T61722 CYN7X3 11690704 IC50 = 0.8 nM T61722 C9CM2R 11695689 IC50 = 15 nM T61722 CH40CJ 11696710 IC50 = 29 nM T61722 CL1F3A 11697751 IC50 = 3.6 nM T61722 CULM38 11704178 IC50 = 1.3 nM T61722 CG97HW 11704605 IC50 = 30 nM T61722 CT36JS 11704767 IC50 = 1.5 nM T61722 CNJ1V5 11709353 Ki = 504 nM T61722 C8JT3C 11709441 Ki = 270 nM T61722 CZTE59 11717304 IC50 = 7 nM T61722 C4AS6M 11717784 Ki = 299 nM T61722 COSR23 11717904 Ki = 158 nM T61722 CTR93A 11718652 Ki = 23 nM T61722 C4EX2F 11742188 IC50 = 23 nM T61722 CFX9G7 11818138 IC50 = 178 nM T61722 CCB54R 12341157 Ki > 10000 nM T61722 CSJ4D1 13507348 IC50 = 165 nM T61722 CD7V5E 15422467 IC50 = 560 nM T61722 C4TN7A 15948907 Ki = 1660 nM T61722 C3X8SB 15949007 Ki = 758 nM T61722 CQSU29 15949201 Ki = 960 nM T61722 C2KM0C 15949202 Ki = 1759 nM T61722 C0V6OT 15949299 Ki = 36 nM T61722 CR0O9U 15949300 Ki = 143 nM T61722 CAZ41C 15949301 Ki = 233 nM T61722 CIA53V 15949302 Ki = 1506 nM T61722 CI9SU8 15949395 Ki = 10 nM T61722 C2ZM3S 15949483 Ki = 596 nM T61722 CUYG13 15949576 Ki = 51 nM T61722 C0AE7Y 15949577 Ki = 1338 nM T61722 CH81IN 15949578 Ki = 497 nM T61722 C89SAY 15949579 Ki = 12 nM T61722 CWD64O 15949676 Ki = 1536 nM T61722 CHBE61 15949677 Ki = 23 nM T61722 C4NUX3 15949678 Ki = 870 nM T61722 CNY93T 15949679 Ki = 1172 nM T61722 C7H8AT 15949759 Ki = 438 nM T61722 C7BT4J 15949760 Ki = 1300 nM T61722 CUJ30Y 15949761 Ki = 318 nM T61722 C3AQY9 15949762 Ki = 43 nM T61722 C8KI4N 15949763 Ki = 21 nM T61722 C5N0UZ 15949764 Ki = 25 nM T61722 C52FLP 15949765 Ki = 37 nM T61722 C87TMW 15949849 Ki = 89 nM T61722 C5RB1S 15949851 Ki = 154 nM T61722 CIQ9M2 15949852 Ki = 20 nM T61722 CG42RP 15950020 Ki = 38 nM T61722 CKS79G 15950100 Ki = 68 nM T61722 CHV69J 15950102 Ki = 37 nM T61722 CCAQ82 15950103 Ki = 96 nM T61722 CCJA08 15950184 Ki = 115 nM T61722 CLB1V3 15950186 Ki = 169 nM T61722 C79VQK 15950271 IC50 = 156 nM T61722 CMY2A4 15950273 Ki = 356 nM T61722 CTM05L 15950274 Ki = 267 nM T61722 CB7F2R 15950276 Ki = 747 nM T61722 C0NQV6 16093474 Ki = 28 nM T61722 C0F5XY 16118987 IC50 = 3.1 nM T61722 C20DXZ 16222206 IC50 = 4.8 nM T61722 CRZT49 16222207 IC50 = 0.012 nM T61722 C5Z3EJ 16660132 IC50 = 15 nM T61722 CGF9A8 16660133 IC50 = 0.46 nM T61722 CC8QP4 16660134 IC50 = 2 nM T61722 CHMZ19 16660287 IC50 = 1.5 nM T61722 CNA70H 16660288 IC50 = 0.24 nM T61722 C96URO 16660289 IC50 = 4.4 nM T61722 CP49ZE 16660290 IC50 = 0.072 nM T61722 CK6Q9V 16660291 IC50 = 15 nM T61722 CQGL62 16678407 IC50 = 79 nM T61722 CPV0C8 16678600 IC50 = 11 nM T61722 C5PK9I 16678601 IC50 = 2.2 nM T61722 CAE4V0 16678606 IC50 = 50 nM T61722 CFQ7J5 17121284 IC50 = 5500 nM T61722 C2D1QF 21093095 IC50 = 217 nM T61722 CC40FD 22935741 IC50 = 200 nM T61722 CBD49O 22935743 IC50 = 540 nM T61722 CM9I4A 23582349 Ki = 1060 nM T61722 C1ML6Y 23582350 Ki = 2940 nM T61722 CF81SW 23582412 IC50 = 0.4 nM T61722 C4Y5WB 23634381 Ki = 32 nM T61722 CM4HU9 23661689 Ki = 0.631 nM T61722 CXTU69 23725171 IC50 = 5 nM T61722 CI1G4X 23800745 IC50 = 2400 nM T61722 CSBT13 24743756 Ki < 1000 nM T61722 C42LYP 24765153 Ki = 233 nM T61722 CF72YI 24765671 Ki >= 785 nM T61722 C31JZP 24765672 Ki >= 2500 nM T61722 C4QX7Y 24765675 Ki >= 930 nM T61722 CL7Z9U 24765768 Ki >= 110 nM T61722 C8NVE5 24776278 Ki = 712 nM T61722 C5FCS8 24776279 Ki = 2741 nM T61722 C9Y0NH 24776280 Ki > 30000 nM T61722 CR9XD6 24776281 Ki = 4669 nM T61722 CUJA73 24776282 Ki = 3829 nM T61722 CG9BL8 24776283 Ki = 769 nM T61722 C8VYO3 24776284 Ki = 11629 nM T61722 CI9O6X 24776285 Ki = 7615 nM T61722 C2D0KF 24776286 Ki = 1448 nM T61722 C36COI 24776287 Ki = 8903 nM T61722 C8HSU4 24776288 Ki = 4131 nM T61722 CB1Z9P 24776289 Ki = 4174 nM T61722 CTW27D 24776290 Ki > 30000 nM T61722 C85KOC 24776291 Ki = 24 nM T61722 CUMH30 24776292 Ki = 55 nM T61722 CNT80M 24776293 Ki = 212 nM T61722 CVR6K5 24776294 Ki = 7.6 nM T61722 CU1S4P 24776295 Ki = 5.3 nM T61722 CJC64I 24776296 Ki = 702 nM T61722 CAME19 24776297 Ki = 32 nM T61722 CFX7T3 24776298 IC50 = 0.23 nM T61722 CE3Q0W 24776299 Ki = 2200 nM T61722 CED0V5 24776300 Ki = 81 nM T61722 CG9PI2 24776301 Ki = 2044 nM T61722 CLS5J9 24776302 Ki = 23 nM T61722 CEBZ45 24776303 Ki = 926 nM T61722 C8GRM0 24776304 IC50 = 18 nM T61722 CFYH26 24776305 Ki = 302 nM T61722 C4BD1L 24776306 Ki = 5.3 nM T61722 CMJ2P1 24776307 Ki = 13 nM T61722 CD42AZ 24776308 Ki = 13 nM T61722 CFQA40 24952577 Ki > 7282 nM T61722 CD98IN 24952580 Ki > 456 nM T61722 C81WVN 24952927 Ki > 5474 nM T61722 CZT83E 24952928 Ki > 501 nM T61722 C8YHX3 24953283 Ki > 224 nM T61722 CZ93FO 24953285 Ki > 628 nM T61722 C17JTY 24953286 Ki > 2226 nM T61722 CFT0W5 24953624 Ki > 4992 nM T61722 C42VMD 24953625 Ki > 3461 nM T61722 C7B2EW 24953628 Ki > 2117 nM T61722 C05VGF 24961406 IC50 = 42 nM T61722 CPX1U2 24962860 IC50 = 18 nM T61722 CIE9K4 24995212 Ki = 5.4 nM T61722 CXQJ67 25002382 Ki >= 1291 nM T61722 CN5SH9 25003075 Ki > 21000 nM T61722 CDR8B5 25106870 IC50 = 220 nM T61722 CQSC30 25106871 IC50 = 22 nM T61722 CEX34J 25817650 Ki = 0.6 nM T61722 CO46CI 25908688 Ki = 2250 nM T61722 CG9F0D 25908691 Ki = 75 nM T61722 C0TF5X 29264684 IC50 = 2100 nM T61722 CF1EL0 39200227 IC50 = 520 nM T61722 CB0UH5 39453523 IC50 = 860 nM T61722 C4EI6R 39453527 IC50 = 1500 nM T61722 CZG4X7 44128594 IC50 = 9 nM T61722 CNOF71 44138108 Ki = 4789 nM T61722 CFM7Y4 44158600 IC50 = 7 nM T61722 CJM81I 44158825 IC50 = 1 nM T61722 CW2D9F 44158941 IC50 = 5 nM T61722 CHP52S 44158942 IC50 = 12 nM T61722 CF97PS 44159058 IC50 = 8 nM T61722 C5G4LN 44159411 IC50 = 8 nM T61722 CUEC20 44159529 IC50 = 18 nM T61722 CHI65U 44159530 IC50 = 5 nM T61722 CI32KG 44159646 Ki = 13.5 nM T61722 C2SQJ7 44159647 IC50 = 4 nM T61722 CGT5Z8 44159648 IC50 = 10 nM T61722 CF59OP 44159650 IC50 = 29 nM T61722 CSG9M6 44159769 IC50 = 7 nM T61722 C5UBJ4 44159770 IC50 = 3 nM T61722 CA8L9H 44159771 IC50 = 4 nM T61722 CMNH53 44159772 IC50 = 3 nM T61722 C9FQT1 44159773 IC50 = 2 nM T61722 CUE81M 44188793 IC50 = 90 nM T61722 C48ZIW 44188794 IC50 = 2750 nM T61722 CISJ51 44188797 IC50 = 1130 nM T61722 C0FN6X 44188965 IC50 = 1630 nM T61722 CXV97L 44188966 IC50 = 230 nM T61722 C0D9FV 44188967 IC50 = 390 nM T61722 C7AGZ4 44189135 IC50 = 3000 nM T61722 CKB32S 44189138 IC50 = 4000 nM T61722 CW50TD 44195251 IC50 = 53 nM T61722 CLG9O7 44205512 IC50 = 880 nM T61722 C6WTU0 44205513 IC50 = 360 nM T61722 C5G4NL 44205514 IC50 = 1300 nM T61722 CCPI98 44205720 IC50 = 340 nM T61722 CZ29JY 44205724 IC50 = 180 nM T61722 CJ9Q2B 44207788 IC50 = 45 nM T61722 C7P8OX 44249133 IC50 = 3.981 nM T61722 C7GN8J 44390215 Ki = 3000 nM T61722 CIO51Y 44390216 Ki = 33000 nM T61722 CF2IU0 44390221 Ki = 3300 nM T61722 C34RSB 44390224 Ki = 27000 nM T61722 CEJX46 44390242 Ki = 30 nM T61722 CAZY30 44390248 Ki = 7500 nM T61722 CQM97O 44390249 Ki = 4400 nM T61722 C0NIT4 44390259 Ki = 2100 nM T61722 CJD3N8 44390264 Ki = 18000 nM T61722 C8EG2Q 44390268 Ki = 250 nM T61722 C9SJ1O 44390269 Ki > 50000 nM T61722 CI51GJ 44390270 Ki = 7400 nM T61722 C0QXS8 44390275 Ki = 17000 nM T61722 C3RWO1 44390276 IC50 = 130 nM T61722 CX4KY0 44390277 Ki = 8300 nM T61722 C0W4ZJ 44390287 Ki = 1300 nM T61722 CPLU35 44390288 Ki > 50000 nM T61722 CH6MN2 44390290 Ki = 7400 nM T61722 CLO32H 44390292 Ki = 2400 nM T61722 CESG92 44390294 Ki = 4600 nM T61722 C8NY4U 44390298 Ki = 1700 nM T61722 C9O0FJ 44390303 Ki = 6400 nM T61722 C6JZ1L 44390305 Ki = 970 nM T61722 C6MAW3 44390306 Ki = 1200 nM T61722 CNGD14 44390311 Ki > 50000 nM T61722 C9MAN2 44390312 Ki = 20 nM T61722 CZNS52 44390316 Ki = 3600 nM T61722 C3X5RM 44390318 Ki = 3200 nM T61722 C53SFI 44390324 Ki = 19000 nM T61722 CI41SJ 44390327 Ki = 4200 nM T61722 CBS0A1 44390328 Ki = 4200 nM T61722 CA0D1C 44390331 Ki > 50000 nM T61722 CDO76V 44390332 IC50 = 22 nM T61722 CAS25H 44390333 Ki > 50000 nM T61722 C0X9ZM 44390342 Ki > 50000 nM T61722 CNP29E 44390343 Ki = 7600 nM T61722 CIX8C9 44390348 Ki > 50000 nM T61722 CJR48Z 44390350 Ki > 50000 nM T61722 CJKM84 44390354 IC50 = 120 nM T61722 CTP1D6 44390930 EC50 = 1.4 nM T61722 CM0E2P 44414678 IC50 = 11 nM T61722 CZO5K3 44414728 IC50 = 50 nM T61722 CWAU29 44414741 IC50 = 125 nM T61722 CB6H5Y 44414758 IC50 = 18 nM T61722 CF2SU8 44414775 IC50 = 68 nM T61722 CU26FW 44414799 IC50 = 5200 nM T61722 CB8KS0 44417446 IC50 = 3.6 nM T61722 C8R7KH 44417453 IC50 = 3.4 nM T61722 C0XVJ1 44417456 IC50 = 391 nM T61722 CSH6T9 44417459 IC50 = 5350 nM T61722 CV0D3X 44417460 IC50 = 108 nM T61722 C4QR8I 44417462 IC50 = 48 nM T61722 CW2D9I 44417463 IC50 = 151 nM T61722 CG3E7T 44417465 IC50 = 47 nM T61722 C8JW7Z 44417467 IC50 = 42 nM T61722 CCN27R 44417469 IC50 = 37 nM T61722 C1JGY7 44417474 IC50 = 13 nM T61722 CND06K 44441186 Ki > 10000 nM T61722 C1OKM8 44441196 Ki = 90 nM T61722 CRA6S0 45109984 Ki = 21.1 nM T61722 C3JE7N 45109987 IC50 = 2.3 nM T61722 CA28PL 45109988 IC50 = 7 nM T61722 CN6P8B 45109989 IC50 = 4.4 nM T61722 CY2BK4 45110108 Ki = 3.4 nM T61722 CR1KP4 45110109 IC50 = 3.4 nM T61722 CR6UW4 45112038 IC50 = 1.2 nM T61722 CULJ91 45268456 IC50 = 94 nM T61722 CY0H3M 45268524 IC50 = 18 nM T61722 CB5O6V 45269307 IC50 = 4 nM T61722 C03ETI 45270148 IC50 = 457 nM T61722 CJ42OZ 45270214 Ki = 1171 nM T61722 CY70SI 45270983 IC50 = 6 nM T61722 C2XH3A 45270987 IC50 = 860 nM T61722 C35DUQ 45272700 IC50 = 18 nM T61722 CKUI32 45272704 IC50 = 96 nM T61722 C6BV0R 45272761 IC50 = 5 nM T61722 CM26PO 45273621 Ki = 35 nM T61722 C3U7KT 45273637 Ki = 7189 nM T61722 C4XE5C 45486009 IC50 = 7 nM T61722 CUBP04 45486015 IC50 = 3 nM T61722 CN5XU9 45486016 IC50 = 680 nM T61722 C1N8TO 45486017 IC50 = 1400 nM T61722 C0L5AY 45486021 IC50 = 4 nM T61722 C3Y7KG 45486025 IC50 = 107 nM T61722 C2UZP0 45486026 IC50 = 4 nM T61722 CJ6QF2 45486029 IC50 = 4 nM T61722 CR7YG5 45486030 IC50 = 3 nM T61722 C0WR7I 45486034 IC50 = 130 nM T61722 C14LAV 45486038 IC50 = 6 nM T61722 CQG87L 45486039 IC50 = 4 nM T61722 CU56JW 45486040 IC50 = 7 nM T61722 CLO03H 45486043 IC50 = 4.7 nM T61722 CZ6JL3 45486044 IC50 = 47 nM T61722 CE3V7H 45486045 IC50 > 50000 nM T61722 CAD20G 45486052 IC50 = 7 nM T61722 CX0AO7 45486053 IC50 = 2370 nM T61722 C1YRG8 45486054 IC50 = 2 nM T61722 CSX4B2 45486056 IC50 = 12 nM T61722 CGB8C5 45486057 IC50 = 3 nM T61722 CR4NA1 45486058 IC50 = 1100 nM T61722 CHK46L 45486059 IC50 = 740 nM T61722 CGJ5A6 45486064 IC50 = 16 nM T61722 CD6XC5 45486065 IC50 = 2 nM T61722 CYI19K 45486071 IC50 = 5 nM T61722 C2ZO7I 45486072 IC50 = 28 nM T61722 CK4ZB3 45486073 IC50 = 16 nM T61722 CF24XK 45486074 IC50 = 2 nM T61722 CH58TM 45486094 IC50 = 13 nM T61722 CV6RL2 45486095 IC50 = 380 nM T61722 CYW91F 45486098 IC50 > 10000 nM T61722 C7QEA3 45486099 IC50 = 2 nM T61722 CRCS08 45486100 IC50 = 3 nM T61722 C5W4RK 46189872 IC50 = 0.02 nM T61722 C54DMW 46216756 IC50 = 3.7 nM T61722 C6PVJ9 46229750 IC50 = 40 nM T61722 C2A5IB 46229751 IC50 = 18 nM T61722 CY41FX 46229752 IC50 = 14 nM T61722 CWYJ86 46229753 IC50 = 16 nM T61722 CG3S8R 46229758 IC50 = 1800 nM T61722 CJ86TZ 46229759 IC50 = 3800 nM T61722 C7LIV4 46229760 IC50 = 140 nM T61722 C2ASY9 46229761 IC50 = 700 nM T61722 C7OSC9 46229762 IC50 = 24 nM T61722 C5VG6R 46229798 IC50 = 1300 nM T61722 C14JFY 46229799 IC50 = 3300 nM T61722 CAGX74 46229800 IC50 = 510 nM T61722 CX08EY 46229801 IC50 = 5.3 nM T61722 CN67KW 46229805 IC50 = 510 nM T61722 CX98KO 46229806 IC50 = 170 nM T61722 CP9K2Q 46229807 IC50 = 340 nM T61722 CL1V8X 46229808 IC50 = 270 nM T61722 C4KGT8 46229845 IC50 = 0.48 nM T61722 CED2I9 46229846 IC50 = 3.1 nM T61722 C1DK4I 46229847 IC50 = 110 nM T61722 C9EQ4H 46229852 IC50 = 40 nM T61722 C1FUD8 46229853 IC50 = 170 nM T61722 C8UHT3 46229854 IC50 = 160 nM T61722 C97JVD 46229855 IC50 = 24 nM T61722 CEA65M 46229883 IC50 = 3800 nM T61722 C95GXW 46229884 IC50 = 380 nM T61722 CJLM59 46229885 IC50 = 890 nM T61722 C2JCI8 46229886 IC50 = 220 nM T61722 CBC8P9 46229890 IC50 = 160 nM T61722 C7YXM2 46229891 IC50 = 41 nM T61722 COGB82 46229936 IC50 = 180 nM T61722 CY2D1N 46229937 IC50 = 190 nM T61722 C8MT4K 46229938 IC50 = 2900 nM T61722 CQYG70 46229939 IC50 = 52 nM T61722 C9IHO6 46229940 IC50 = 25 nM T61722 CO7L6Y 46229941 IC50 = 380 nM T61722 CDO0L8 46229942 IC50 = 660 nM T61722 CPA95T 46229943 IC50 = 230 nM T61722 CN0E1R 46229989 IC50 = 390 nM T61722 CV5A7Q 46229990 IC50 = 450 nM T61722 CFJ5Q2 46229991 IC50 = 360 nM T61722 CQDW60 46229992 IC50 = 500 nM T61722 C8E3MK 46229993 IC50 = 880 nM T61722 CF12XE 46229994 IC50 = 71 nM T61722 C72XQO 46230041 IC50 = 730 nM T61722 CZ4F9C 46230042 IC50 = 32 nM T61722 C41CDK 46230043 IC50 = 2000 nM T61722 C0E6VL 46230044 IC50 = 570 nM T61722 C9BWK1 46230091 IC50 = 93 nM T61722 CYL67Q 46230092 IC50 = 340 nM T61722 CFI9L1 46230093 IC50 = 56 nM T61722 CCPQ30 46230147 IC50 = 530 nM T61722 C0PQ4Y 46230148 IC50 = 17 nM T61722 C23XNK 46230186 IC50 = 9.7 nM T61722 CR12HW 46230187 IC50 = 810 nM T61722 C5X8QZ 46230188 IC50 = 61 nM T61722 CA4FU5 46230191 IC50 = 38 nM T61722 C9PX8L 46230225 IC50 = 3200 nM T61722 C2I9XC 46230227 IC50 = 16 nM T61722 CKO8L9 46230233 IC50 = 820 nM T61722 CM68TS 46230234 IC50 = 160 nM T61722 C9P2LH 46230235 IC50 = 470 nM T61722 CTUA65 46230282 IC50 = 910 nM T61722 C43PVH 46230283 IC50 = 1100 nM T61722 C2J4UR 46230284 IC50 = 9400 nM T61722 CW3S1V 46230289 IC50 = 660 nM T61722 C4NOH8 46230331 IC50 > 100000 nM T61722 CN0O4G 46230336 IC50 = 310 nM T61722 C7BR8E 46230337 IC50 = 940 nM T61722 C3NV2L 46230375 IC50 = 3.4 nM T61722 C5JM7Y 46230380 IC50 = 700 nM T61722 CY75SQ 46230381 IC50 = 1200 nM T61722 C8Z4HO 46230423 IC50 = 35 nM T61722 C29ICH 46230424 IC50 = 150 nM T61722 C8I4CN 46230425 IC50 = 20 nM T61722 CS69ZI 46230430 IC50 = 220 nM T61722 C93GSX 46230511 IC50 = 57 nM T61722 CEV6W5 46230512 IC50 = 1500 nM T61722 C31ARD 46230513 IC50 = 140 nM T61722 C0A8IT 46230514 IC50 = 590 nM T61722 C1VN0G 46230519 IC50 = 94 nM T61722 CLT34W 46230520 IC50 = 88 nM T61722 C2GY5B 46230521 IC50 = 220 nM T61722 CP0TJ8 46230522 IC50 = 360 nM T61722 C6RV7G 46701878 IC50 = 13 nM T61722 C90NLX 46853755 Ki = 2 nM T61722 C5YFG3 46865091 Ki = 41 nM T61722 CR86WT 46865196 Ki = 43 nM T61722 CD15SZ 46865197 Ki = 14 nM T61722 C3U6CI 46865198 Ki = 16 nM T61722 CGOZ93 46865200 Ki = 3.5 nM T61722 C8R1MJ 46865201 Ki = 44 nM T61722 CE79RH 46865310 Ki = 1.3 nM T61722 CZ2V6S 46865311 Ki = 12 nM T61722 CBJ30P 46865312 Ki = 23 nM T61722 CD7EB5 46865413 Ki = 25 nM T61722 C92NKP 46865414 Ki = 14 nM T61722 CFR86P 46865523 Ki = 65 nM T61722 C5CWI2 46865524 Ki = 57 nM T61722 CH7E6U 46865759 Ki = 1470 nM T61722 C6E8GM 46865760 Ki = 60 nM T61722 C6ASU9 46865761 Ki = 28 nM T61722 C2P0SC 46865762 Ki = 29 nM T61722 C2Q3LH 46865763 Ki = 47 nM T61722 CJY7L5 46865873 Ki = 1120 nM T61722 CKO15S 46865874 Ki = 9 nM T61722 CL28XJ 46865875 Ki = 183 nM T61722 CAP4Z1 46865879 Ki = 28 nM T61722 CC1HB5 46865969 Ki = 22 nM T61722 CY69PE 46865970 Ki = 19 nM T61722 C57AHQ 46865971 Ki = 12 nM T61722 CN4IF0 46865973 Ki = 6 nM T61722 CLN24P 46865974 Ki = 4 nM T61722 C1MQ4Y 46866072 Ki = 72 nM T61722 C2O5WU 46866074 Ki = 3.5 nM T61722 CMWG79 46866175 Ki = 14 nM T61722 CAV1Q7 46866265 Ki = 12 nM T61722 CPJ0O8 46866266 Ki = 5 nM T61722 C6L0TD 46866267 Ki = 10 nM T61722 CF34DY 46866268 Ki = 5 nM T61722 CBK07M 46866269 Ki = 5 nM T61722 CFH2K8 46866270 Ki = 86 nM T61722 C31JSK 46866377 Ki = 65 nM T61722 C7Y3VS 46866378 Ki = 2.9 nM T61722 CY2DM8 46866381 Ki = 3.1 nM T61722 CS24CG 46866382 Ki = 4.1 nM T61722 CBFN73 46866480 Ki = 6 nM T61722 C4U5QC 46866481 Ki = 4.2 nM T61722 CLO63K 46866583 Ki = 3.6 nM T61722 C5TF8Q 46866585 Ki = 287 nM T61722 CBJ2C5 46866588 Ki = 369 nM T61722 C12CAY 46866688 Ki = 55 nM T61722 CD42HA 46866690 Ki = 52 nM T61722 CCJ85N 46878930 IC50 = 1420 nM T61722 CS4W5J 46878931 IC50 = 910 nM T61722 CG12CM 46878981 IC50 = 3170 nM T61722 C4ZY7F 46879022 IC50 = 5 nM T61722 CD79OA 46879023 IC50 = 29 nM T61722 C9U7SC 46879131 IC50 = 22 nM T61722 CC7HW8 46879132 IC50 = 2280 nM T61722 CY14RC 46879133 IC50 = 40300 nM T61722 C4M2SQ 46879190 IC50 = 250 nM T61722 C5O2FY 46879283 IC50 = 62000 nM T61722 C27BNS 46879284 IC50 = 74 nM T61722 CEK1D8 46879285 IC50 = 41 nM T61722 C6X9QA 46879286 IC50 = 92 nM T61722 COD7B2 46879319 IC50 = 26 nM T61722 C8DPY5 46879342 IC50 = 13 nM T61722 C2L3DI 46879343 IC50 = 0.77 nM T61722 C2T4RS 46879344 IC50 = 39 nM T61722 CI3RS4 46879377 IC50 = 25 nM T61722 CRS2A6 46880246 IC50 > 100 nM T61722 CC41WH 46880247 IC50 > 100 nM T61722 CWQ98D 46880900 IC50 = 0.085 nM T61722 CN72GY 46880901 IC50 = 75 nM T61722 CZ3A9E 46880939 IC50 = 0.2 nM T61722 CKBT02 46880940 IC50 = 9140 nM T61722 CD2S6V 46880941 IC50 = 2070 nM T61722 CVL0A6 46890028 Ki = 1500 nM T61722 CFQC07 46890029 Ki = 690 nM T61722 CU2YI8 46890030 Ki = 430 nM T61722 C8D4YX 46890031 Ki = 8100 nM T61722 C4Y6JS 46890032 Ki = 2300 nM T61722 C4S6KN 46890086 Ki = 1100 nM T61722 CL6NS3 46890087 Ki = 630 nM T61722 C8NP5C 46890088 Ki = 18 nM T61722 C8JG5T 46890089 Ki = 560 nM T61722 CPQ04X 46890134 Ki = 920 nM T61722 CCT2V9 46890135 Ki = 480 nM T61722 CZT6Y9 46890136 Ki = 12 nM T61722 CI5MX3 46890137 Ki = 13 nM T61722 CUB7X2 46890177 Ki = 8 nM T61722 C7XUP2 46890178 Ki = 220 nM T61722 CA4LM0 46890179 Ki = 29 nM T61722 CZ6OK4 46890180 Ki = 35 nM T61722 C6RBS5 46890208 Ki = 1400 nM T61722 CX5VP4 46890209 Ki = 1400 nM T61722 C0A2CI 46890616 Ki >= 504 nM T61722 CW52VH 46890658 Ki >= 260 nM T61722 CXQ2W0 46890659 Ki >= 580 nM T61722 CQ20RC 46890660 Ki >= 100 nM T61722 C6P1IW 46890683 Ki = 9200 nM T61722 CP34ZN 46890684 Ki = 2900 nM T61722 C2L9KW 46890685 Ki = 2900 nM T61722 C6XS1G 46890686 Ki = 2000 nM T61722 CN9GF0 46890687 Ki = 2800 nM T61722 C8U9SL 49765145 Ki = 108 nM T61722 C3DN7U 49843520 Ki = 5.7 nM T61722 CCX18D 49871902 Ki = 3.1 nM T61722 CL7U6H 49871904 Ki = 56 nM T61722 CXI9D0 49871995 Ki = 26 nM T61722 CV29RM 49872188 Ki = 5.2 nM T61722 CQ30GI 49872288 Ki = 2.2 nM T61722 C3Y6NV 49872386 Ki = 140 nM T61722 CXM42Y 49872387 Ki = 10 nM T61722 CPM08K 49872388 Ki = 39 nM T61722 CLQB36 49872390 Ki = 18 nM T61722 C2ZG9D 49872391 Ki = 7 nM T61722 CJ1MC0 49872486 Ki = 5.6 nM T61722 CHL02B 49872487 Ki = 11 nM T61722 CPUY61 49872488 Ki = 3.3 nM T61722 CR8AC1 49872489 Ki = 45 nM T61722 C1YZ7L 49872490 Ki = 7.1 nM T61722 C2UT4S 49872580 Ki = 44 nM T61722 C43QJD 49872582 Ki = 12 nM T61722 CS47WU 49872583 Ki = 50 nM T61722 CLBO38 49872584 Ki = 620 nM T61722 CF10ZE 49872586 Ki = 42 nM T61722 CO0Y6K 49872677 Ki = 110 nM T61722 C2W6TX 49872682 Ki = 360 nM T61722 CZ6J4P 49872683 Ki = 220 nM T61722 CJWE29 49872771 Ki = 220 nM T61722 CK9VE4 49872772 Ki = 4.5 nM T61722 CYUG08 49872773 Ki = 1800 nM T61722 C2MRS9 49872774 Ki = 1200 nM T61722 C7DET4 49872775 Ki = 1400 nM T61722 CJ7IU8 49872776 Ki = 950 nM T61722 C1CMS5 49872777 Ki = 130 nM T61722 CFP14Q 49872867 Ki = 7.7 nM T61722 C83CTW 49872868 Ki = 6.9 nM T61722 C5EHW3 49872869 Ki = 3 nM T61722 CB41UE 49872870 Ki = 3 nM T61722 CN5JV9 49872871 Ki = 8.2 nM T61722 CLB34U 49872872 Ki = 19 nM T61722 CI2UV5 49872960 Ki = 7.6 nM T61722 CDK4P8 49872965 Ki = 3.6 nM T61722 CAM1D0 49873181 Ki = 2.4 nM T61722 CVE57H 49873273 Ki = 69 nM T61722 CY86XC 49873366 Ki = 580 nM T61722 CY7QF8 49873368 Ki = 6.4 nM T61722 CM06FG 50898361 Ki > 7230 nM T61722 CZ9UD6 50901657 IC50 = 1.7 nM T61722 CT3K2H 50902400 Ki = 260 nM T61722 C2EJT7 50902473 Ki = 110 nM T61722 C8VNM2 51003549 Ki = 3.3 nM T61722 COZ42H 51031012 IC50 = 13 nM T61722 C9UO5T 51347010 IC50 = 31000 nM T61722 CVCQ34 51347011 IC50 = 50 nM T61722 CN80GS 51347012 IC50 = 10 nM T61722 C6Z7LM 51356842 IC50 = 100 nM T61722 CS65EJ 51357123 IC50 = 28 nM T61722 CJ60LU 51357124 IC50 = 9 nM T61722 C61DQW 51357125 IC50 = 0.3 nM T61722 C1BF3J 51357126 IC50 = 20 nM T61722 C3RPO7 51357127 IC50 = 1.3 nM T61722 C3MLR1 51357128 IC50 = 708 nM T61722 CH2G0D 52918794 IC50 = 90 nM T61722 C0N1VL 52918912 IC50 = 934 nM T61722 CE7ZS9 52918913 IC50 = 104 nM T61722 C98XLP 52919028 IC50 = 4 nM T61722 CF2GU1 52919029 IC50 = 8 nM T61722 CT7Y6U 52919030 IC50 = 137 nM T61722 CYAR16 52919031 IC50 = 0.8 nM T61722 C71JCH 52919156 IC50 = 8 nM T61722 C3PXZ4 52919158 IC50 = 4 nM T61722 CBN4K9 52919280 IC50 = 7 nM T61722 CTQM96 52919413 IC50 = 3 nM T61722 C26POW 52919415 IC50 > 1000 nM T61722 C29KEF 52919417 IC50 > 1000 nM T61722 C2I5EV 52919547 IC50 > 1000 nM T61722 C9F6WT 52919549 IC50 > 1000 nM T61722 CMYN39 52919551 IC50 = 150 nM T61722 C7H8LU 52919670 IC50 > 1000 nM T61722 C0Q4WS 52919672 IC50 = 4 nM T61722 CB6S2Q 52920034 IC50 = 10 nM T61722 CUKQ38 52920145 IC50 = 32 nM T61722 C8JO5D 52920146 IC50 = 16 nM T61722 C0WX6K 52920147 IC50 = 15 nM T61722 C9TL4G 52920150 IC50 = 16 nM T61722 CGUS75 52920262 IC50 = 29 nM T61722 CJD25G 52920263 IC50 = 0.8 nM T61722 CB16OE 52920267 IC50 = 192 nM T61722 CLE89N 52920390 IC50 = 1000 nM T61722 C17LSO 52920391 IC50 = 123 nM T61722 CNZ73K 52920392 IC50 = 107 nM T61722 C2AUL9 53248760 Ki = 1.8 nM T61722 CP3J9M 53248845 IC50 = 3 nM T61722 CTU93P 53316532 Ki = 6725 nM T61722 C4P2CV 53316653 Ki = 8.8 nM T61722 CS4G5H 53316671 Ki = 2.5 nM T61722 CL96IZ 53316672 Ki = 7.6 nM T61722 CBT1P4 53316673 Ki = 117 nM T61722 CMH51O 53317503 IC50 = 201 nM T61722 C8D7UQ 53317569 Ki = 3.7 nM T61722 C1CFU7 53317642 IC50 = 250 nM T61722 CXV3W2 53317718 Ki = 1.4 nM T61722 C0ZH3X 53317854 Ki = 3.6 nM T61722 CP14EK 53317957 Ki = 1.1 nM T61722 C97LDX 53317958 Ki = 1.1 nM T61722 C5WO9J 53317977 Ki = 4.3 nM T61722 C6L0YQ 53318324 IC50 = 1800 nM T61722 COJ82D 53319320 Ki = 1 nM T61722 C4T9BV 53319321 Ki = 1.8 nM T61722 CE86AP 53319322 Ki = 4.4 nM T61722 CO0YD9 53319673 IC50 = 1300 nM T61722 CV8M5K 53320594 Ki = 144 nM T61722 CZL85A 53320595 IC50 = 3 nM T61722 C8EO2U 53320616 Ki = 2.4 nM T61722 C5HY9K 53320617 Ki = 1.6 nM T61722 CZ40CV 53320618 Ki = 6.3 nM T61722 CIU6E0 53321678 IC50 = 15 nM T61722 C7D5BN 53321784 Ki = 139 nM T61722 C5QOI8 53321785 Ki = 1.8 nM T61722 CS2YH5 53321815 IC50 = 3 nM T61722 CZ9O8L 53321816 IC50 = 9 nM T61722 C89DLV 53321923 IC50 = 24 nM T61722 C29QNI 53321924 Ki = 5.5 nM T61722 CJ7C4U 53321925 Ki = 20 nM T61722 C45FQB 53322311 IC50 = 1500 nM T61722 CB5S0H 53322785 Ki = 3.7 nM T61722 CSL4X3 53323125 IC50 = 7 nM T61722 CGA5Z7 53323126 IC50 = 27 nM T61722 CPI3O6 53323246 Ki = 11 nM T61722 C2KRB3 53323266 Ki = 4 nM T61722 CMK0A1 53323267 IC50 = 1.6 nM T61722 C4ZP8Y 53323268 Ki = 4.9 nM T61722 CV3X9R 53323666 IC50 = 190 nM T61722 CTOY32 53324111 Ki = 40.8 nM T61722 CE23YH 53324462 Ki = 1.9 nM T61722 CF9SZ3 53324589 Ki = 1.7 nM T61722 C1RB5O 53324951 IC50 = 330 nM T61722 CC3WP1 53324952 IC50 = 5000 nM T61722 C4H8SB 53325800 IC50 = 27 nM T61722 CUS37X 53325907 IC50 = 5 nM T61722 CZ1SE0 53325908 Ki = 1.6 nM T61722 CH8S3T 53325909 Ki = 17 nM T61722 C9DR3V 53325910 Ki = 21 nM T61722 CZ7WN5 53325911 Ki = 8.7 nM T61722 CEMU31 53325912 IC50 = 63 nM T61722 C5LI8Q 53326243 IC50 = 70 nM T61722 CAL29U 53326879 Ki = 1083 nM T61722 CL89US 53359023 IC50 = 0.9 nM T61722 CZID32 53495002 IC50 = 9 nM T61722 CRB0W3 54580721 Ki = 1.7 nM T61722 CH3RO8 54580742 Ki = 110 nM T61722 CT39WE 54580743 Ki = 19 nM T61722 C5LY7C 54580744 IC50 = 30 nM T61722 C7ZRE2 54580765 IC50 = 36 nM T61722 CTZ14B 54580766 IC50 = 0.1 nM T61722 C2ZNM1 54580767 IC50 = 0.4 nM T61722 C17YIT 54581745 Ki = 370 nM T61722 CI4PB1 54581746 Ki = 1700 nM T61722 C1DRO9 54581747 Ki = 184 nM T61722 CUAI02 54581774 IC50 = 501 nM T61722 CS61FB 54581775 IC50 = 2 nM T61722 CRP57C 54581776 IC50 = 0.2 nM T61722 CF5Y0B 54581777 IC50 = 5650 nM T61722 CB6O3J 54582719 Ki = 340 nM T61722 C9HK6G 54582728 Ki = 15 nM T61722 C7Z3CG 54582729 Ki = 4.3 nM T61722 C2RJM1 54583706 Ki = 7.4 nM T61722 CIYJ59 54583707 Ki = 31 nM T61722 CZ8FO1 54583708 Ki = 408 nM T61722 CC86EI 54583709 Ki = 1220 nM T61722 C5BR0G 54583710 Ki = 3 nM T61722 C1UM6Z 54583731 IC50 = 8912 nM T61722 CKV93Z 54583732 IC50 = 126 nM T61722 CD1YB0 54583733 IC50 = 0.3 nM T61722 C60BSQ 54584664 Ki = 120 nM T61722 C7CME2 54584672 Ki = 240 nM T61722 CGC28Q 54584673 Ki = 70 nM T61722 CP3SG7 54584706 IC50 = 45 nM T61722 C7SXR9 54584707 IC50 = 355 nM T61722 C0RT7L 54584708 IC50 = 178 nM T61722 C65UMA 54584709 IC50 = 3981 nM T61722 C9JW6B 54584710 IC50 = 0.6 nM T61722 C26DVO 54585608 Ki = 14 nM T61722 CZVE41 54585639 IC50 = 251 nM T61722 C8ZH2Q 54585640 IC50 = 0.8 nM T61722 CB0FJ9 54585641 IC50 = 0.2 nM T61722 C5D9TV 54585642 IC50 = 7.9 nM T61722 CB83NJ 54585643 IC50 = 1.6 nM T61722 CJS27M 54585644 IC50 = 891 nM T61722 C7H5SE 54586481 IC50 = 0.2 nM T61722 CBX7L4 54586607 Ki = 141 nM T61722 C6J3IN 54586635 IC50 = 541 nM T61722 CTH6L4 54586636 IC50 = 2.2 nM T61722 CDA35N 54586637 IC50 = 0.6 nM T61722 CVF14M 54586638 IC50 = 0.6 nM T61722 C12IDJ 54587620 Ki = 670 nM T61722 CM75DI 54587621 Ki = 22 nM T61722 C7L9BG 54587622 Ki = 126 nM T61722 CXMJ42 54587623 IC50 = 2 nM T61722 CF2T1P 54587655 IC50 < 0.4 nM T61722 CKHB92 54587656 IC50 = 56 nM T61722 C5V9XF 54587657 IC50 = 10 nM T61722 C8CE3G 54587658 IC50 = 126 nM T61722 CMXZ41 54587659 IC50 = 1.5 nM T61722 CTVF41 54673217 IC50 = 3400 nM T61722 CGC2S9 56589600 Ki = 3.4 nM T61722 CP4B9G 56592488 IC50 = 25 nM T61722 C0RA7C 56594260 Ki = 190 nM T61722 CPX5U9 56594261 Ki = 24 nM T61722 CE36LB 56594262 Ki = 92 nM T61722 CT98IB 56594263 Ki = 101 nM T61722 CPI60V 56594382 Ki = 73 nM T61722 C8U4VP 56594383 Ki = 41 nM T61722 C2R3MJ 56594384 Ki = 117 nM T61722 CAJX90 56594385 Ki = 601 nM T61722 C2JNX8 56594386 Ki = 143 nM T61722 CV7K5G 56594387 Ki = 25 nM T61722 C3LY0B 56594511 Ki = 4.3 nM T61722 CG4RX0 56594512 Ki = 4.9 nM T61722 CJUK12 56594513 Ki = 43 nM T61722 C1WOR8 56594514 Ki = 17 nM T61722 CQ32KJ 56594515 Ki = 15 nM T61722 COX25N 56594516 Ki = 28 nM T61722 CRN31S 56594517 Ki = 10 nM T61722 CUE7F6 56594647 Ki = 5 nM T61722 CFR4Y6 56594648 Ki = 3.3 nM T61722 CTN8C6 56594649 Ki = 8.6 nM T61722 CA1FS4 56594650 Ki = 4.6 nM T61722 C6WKO2 56594651 Ki = 8.6 nM T61722 CA7I9P 56594652 Ki = 3 nM T61722 C27BIS 56594653 Ki = 5 nM T61722 C05MTG 56594779 Ki = 7 nM T61722 C2O3UC 56594780 Ki = 19 nM T61722 CRAH20 56594781 Ki = 8 nM T61722 CW9CQ2 56594782 Ki = 2.1 nM T61722 CY82CA 56594783 Ki = 3.4 nM T61722 C7VYK3 56594784 Ki = 4.4 nM T61722 CE8I1F 56594785 Ki = 3.4 nM T61722 C8AB1G 56594904 Ki = 3.8 nM T61722 C1G5XW 56594905 Ki = 3.6 nM T61722 C7TJ2Z 56594906 Ki = 1.9 nM T61722 CGQ5O0 56594907 Ki = 21 nM T61722 C6A1QC 56594908 Ki = 48 nM T61722 CDG32F 56594909 Ki = 3.2 nM T61722 C50NWY 56594910 Ki = 54 nM T61722 CD9XQ2 56595045 Ki = 122 nM T61722 CY8AB1 56595046 Ki = 60 nM T61722 CK3FG2 56595047 Ki = 37 nM T61722 C82SRT 56595048 Ki = 378 nM T61722 CFY1I0 56595049 Ki = 301 nM T61722 CZT1R5 56595050 Ki = 41 nM T61722 CS7KU1 56595051 Ki = 31 nM T61722 CBIX98 56595181 Ki = 33 nM T61722 CZX8B0 56595182 Ki = 28 nM T61722 CYJ5N1 56595183 Ki = 21 nM T61722 C4H6EZ 56595184 Ki = 25 nM T61722 C5H2OV 56595185 Ki = 5 nM T61722 CKA0S4 56595186 Ki = 7 nM T61722 CAD5R2 56595311 Ki = 8 nM T61722 C2PTH8 56595312 Ki = 46 nM T61722 C47OVL 56595313 Ki = 87 nM T61722 C8K3TR 56595314 Ki = 747 nM T61722 C9KR0G 56595315 Ki = 283 nM T61722 CQ8A9J 56595316 Ki = 4780 nM T61722 CSDG41 56595317 Ki = 55 nM T61722 CUYH89 56595440 Ki = 10 nM T61722 CQ0GX9 56595441 Ki = 24 nM T61722 CS3F0K 56595442 Ki = 21 nM T61722 CAX16V 56595443 Ki = 7 nM T61722 CKGN30 56595569 Ki = 3 nM T61722 CZH1X6 56595570 Ki = 260 nM T61722 C80TZF 56595571 Ki = 1.2 nM T61722 C8J3RV 56595572 Ki = 30 nM T61722 CT2FS7 56595573 Ki = 515 nM T61722 CYN0M9 56643872 IC50 = 22 nM T61722 C7VN2T 56653431 IC50 = 200 nM T61722 C4S5BK 56653781 IC50 = 7.8 nM T61722 C3FL6E 56654115 IC50 = 12 nM T61722 CD32NT 56834987 IC50 = 6 nM T61722 CO65JY 56834988 IC50 > 10000 nM T61722 C6H2JT 56834989 IC50 = 420 nM T61722 CY6UB2 56839590 Ki = 3.2 nM T61722 C1U7XJ 56924869 IC50 = 22 nM T61722 C8NMD9 56924870 IC50 = 24 nM T61722 CIW9Y8 56951184 IC50 = 5.5 nM T61722 C4QJ2R 56959145 Ki = 2.6 nM T61722 CD3AX8 56959274 Ki = 4.7 nM T61722 C2SGE6 56959565 Ki = 1.9 nM T61722 C0QBZ8 56960163 Ki = 7.5 nM T61722 CUF5H4 56960164 Ki = 2.5 nM T61722 C1X5SJ 56960577 Ki = 2.3 nM T61722 CT4SR8 57335620 IC50 = 2 nM T61722 C4BHP5 57335749 IC50 = 8 nM T61722 CA1W8X 57390357 IC50 = 11 nM T61722 CRH1K9 57390757 IC50 = 3 nM T61722 C9BF1I 57390758 IC50 = 5 nM T61722 C8GKR2 57391226 IC50 = 360 nM T61722 CM41FU 57391518 IC50 = 200 nM T61722 CJ5OT4 57391799 IC50 = 15 nM T61722 CI56TU 57391800 IC50 = 3 nM T61722 CN9YJ7 57392165 IC50 = 501 nM T61722 C82IVW 57392166 IC50 = 3.5 nM T61722 C37ERY 57392564 IC50 = 2 nM T61722 CWZ92U 57392565 IC50 = 21 nM T61722 C53WSX 57392566 IC50 = 660 nM T61722 CC9V5H 57392567 IC50 = 400 nM T61722 C3KR1M 57392568 IC50 = 770 nM T61722 C5YCP1 57393037 IC50 = 6.2 nM T61722 C95WXD 57393270 IC50 = 110 nM T61722 C3MXN1 57393532 IC50 = 6 nM T61722 CXR6Y8 57393533 IC50 = 5 nM T61722 CK1ET9 57393918 IC50 = 6.1 nM T61722 CY8ZG3 57393949 Ki = 19 nM T61722 C6ZIH7 57394760 IC50 = 11 nM T61722 C4I9LW 57394761 IC50 = 5.8 nM T61722 C8KY0I 57395006 IC50 = 14 nM T61722 CQ2J9O 57395244 IC50 = 47 nM T61722 C7IL8F 57395245 IC50 = 210 nM T61722 CO8BR1 57395246 IC50 = 5 nM T61722 C7MLC0 57395613 IC50 = 56 nM T61722 C08GIC 57395680 IC50 = 3 nM T61722 C81FYQ 57396042 IC50 = 310 nM T61722 CBR0J8 57396043 IC50 = 10 nM T61722 CQ9OG2 57396044 IC50 = 2 nM T61722 CA23SK 57396512 IC50 = 9.2 nM T61722 C5GBP8 57396745 IC50 > 10000 nM T61722 CDGC05 57396746 IC50 = 350 nM T61722 CW5O7V 57396747 IC50 = 230 nM T61722 CZ1BY9 57396754 IC50 = 76 nM T61722 CFB47P 57396755 IC50 = 15 nM T61722 CSQW63 57396756 IC50 = 2 nM T61722 CP5K2O 57397014 IC50 = 12 nM T61722 C67ZNS 57397461 IC50 = 159 nM T61722 CQ8K7G 57397462 IC50 = 45 nM T61722 C04AJG 57397843 IC50 = 4 nM T61722 C7SW5R 57398275 IC50 = 9800 nM T61722 CV4W9X 57398304 IC50 = 502 nM T61722 C74WUG 57398523 IC50 = 5 nM T61722 CHIB74 57398524 IC50 = 65 nM T61722 C2BLJ3 57398777 IC50 = 5 nM T61722 CD2FV3 57398778 IC50 = 32 nM T61722 CXIN49 57399142 IC50 = 1468 nM T61722 C8I1XR 57399166 Ki = 12 nM T61722 C18FWR 57399938 IC50 = 11000 nM T61722 CO0G1B 57400193 IC50 = 2 nM T61722 CE4VT0 57400453 IC50 = 680 nM T61722 C4DJQ2 57400454 IC50 = 300 nM T61722 C3K7LZ 57400455 IC50 = 7 nM T61722 C3PGK2 57400456 IC50 = 4 nM T61722 C0BFW6 57400457 IC50 = 25 nM T61722 C28QIE 57400864 IC50 = 9.7 nM T61722 CI05FH 57400872 IC50 = 25 nM T61722 CB0F9T 57400908 Ki = 54 nM T61722 C5Q7VD 57401263 IC50 = 6 nM T61722 CFK1Z0 57401719 IC50 = 27000 nM T61722 C0WG9I 57401720 IC50 = 41000 nM T61722 CZHG85 57401747 IC50 = 99 nM T61722 CY0L9P 57401748 IC50 = 17 nM T61722 C3DCU4 57401983 IC50 = 330 nM T61722 CJTF24 57402257 IC50 = 5 nM T61722 CYE63U 57402258 IC50 = 13 nM T61722 C9JS4D 57402607 IC50 = 4 nM T61722 C0AP6W 57402651 IC50 = 89 nM T61722 CY38WL 57402652 IC50 = 1.6 nM T61722 COQ26K 57402653 IC50 = 11 nM T61722 C6YRD9 57402681 Ki = 18 nM T61722 CDJK52 57403006 IC50 = 580 nM T61722 CI68RM 57403987 IC50 = 8 nM T61722 CK76CI 57403988 IC50 = 7 nM T61722 CX13SU 57404015 IC50 = 12 nM T61722 C02JMP 57444239 Ki = 380 nM T61722 CY6PH5 57505154 IC50 = 20 nM T61722 C65LDM 57505183 IC50 = 134 nM T61722 C2A0ZN 57505193 IC50 = 34 nM T61722 C1OY8Q 57505195 IC50 = 0.8 nM T61722 CEVT09 57505196 IC50 = 12 nM T61722 CDNZ76 57505216 IC50 = 135 nM T61722 CTR5W6 57505220 IC50 = 16 nM T61722 C1ZJ7U 57505231 IC50 = 245 nM T61722 CBQ7L8 57505233 IC50 = 76 nM T61722 C7T1JU 57505234 IC50 = 1690 nM T61722 C8ZW9N 57505236 IC50 > 1000 nM T61722 CZPK24 57505238 IC50 = 5 nM T61722 CP7IA0 57505239 IC50 = 7 nM T61722 C6O1AK 57505241 IC50 = 6 nM T61722 C4B0FN 57505242 IC50 = 28 nM T61722 CH1Z4F 57505246 IC50 > 2000 nM T61722 C2ZY3C 57505248 IC50 = 14 nM T61722 C37SMZ 57505249 IC50 = 1.2 nM T61722 CT06AR 57505250 IC50 = 4 nM T61722 C6SJB5 57505254 IC50 = 3 nM T61722 CDY0K6 57505255 IC50 = 18 nM T61722 C68XZM 57505266 IC50 = 42 nM T61722 C9SYN3 57505267 IC50 = 10 nM T61722 CHD35A 57505268 IC50 = 5 nM T61722 CIN0M5 57505270 IC50 = 6 nM T61722 CT67UA 57505271 IC50 = 6 nM T61722 CI89CS 57505273 IC50 = 17 nM T61722 CJA04V 57505278 IC50 = 70 nM T61722 C9P2EI 57505279 IC50 = 195 nM T61722 CFKU45 57505280 IC50 = 711 nM T61722 CWOY32 57505281 IC50 = 84 nM T61722 C28MXF 57505282 IC50 = 148 nM T61722 C1Q0IT 57505286 IC50 = 21 nM T61722 C4RO9X 57505291 IC50 = 8 nM T61722 C4YCN1 57505297 IC50 = 16 nM T61722 C0YF9P 57505298 IC50 = 2000 nM T61722 C7O3KN 57505304 IC50 = 1120 nM T61722 C1JWH2 57505322 IC50 = 23 nM T61722 C7H8TK 57505325 IC50 = 11 nM T61722 CUL3G4 57505332 IC50 = 20 nM T61722 C9TZR5 57505333 IC50 = 2 nM T61722 CI2M8D 57505334 IC50 = 9 nM T61722 CCU0W5 57505335 IC50 = 5 nM T61722 C6XZ0M 57505337 IC50 = 3 nM T61722 C1WX9I 57505338 IC50 = 8 nM T61722 CJ3NS8 57505339 IC50 = 6 nM T61722 C1XCB8 57505341 IC50 = 11 nM T61722 C6YXJ4 57505342 IC50 = 18 nM T61722 CZ1N3I 57505343 IC50 = 11 nM T61722 CNL8A2 57740764 Ki = 19 nM T61722 C41IFE 58017113 Ki = 390 nM T61722 CEAK10 58017115 Ki = 7 nM T61722 C43QAT 58071818 Ki = 0.5 nM T61722 CA84TQ 58071837 Ki = 4.8 nM T61722 CZ75HB 58628171 Ki = 44 nM T61722 CLYM70 59145768 Ki = 0.2 nM T61722 CS85NE 59644621 IC50 = 28 nM T61722 CQ3P6K 59644626 IC50 = 860 nM T61722 C5KZ9N 59644708 IC50 = 5 nM T61722 C4Z9WG 59644732 IC50 = 2510 nM T61722 CK2UL5 59644763 IC50 = 140 nM T61722 C3PO5X 59753850 IC50 = 2 nM T61722 CX4V3U 59864915 IC50 = 8 nM T61722 C7RI1F 60153792 IC50 = 16 nM T61722 CMF3U1 60153793 IC50 > 1000 nM T61722 C45OLU 60153794 IC50 > 1000 nM T61722 C14BRG 60154703 IC50 = 109 nM T61722 C8CRT2 60167966 Ki = 247 nM T61722 C2CKN8 66853624 Ki = 17 nM T61722 C4V1GL 66853825 Ki = 28 nM T61722 CN1M9Y 66853914 Ki = 22 nM T61722 CN7E8B 66853985 Ki = 5.4 nM T61722 C7A2EI 66854102 Ki = 0.9 nM T61722 C9M6ZU 66854780 Ki = 4 nM T61722 CU3LA9 66854874 Ki = 17 nM T61722 CX93PD 66887118 Ki = 2.5 nM T61722 CKLG50 67007255 IC50 = 38 nM T61722 C1I3RW 67007529 IC50 = 36 nM T61722 CIXF85 67007687 IC50 = 210 nM T61722 CD6J9C 67008149 IC50 = 5.2 nM T61722 C1GP6S 67008150 IC50 = 340 nM T61722 CT25QA 67008500 IC50 = 6.1 nM T61722 CW0F9L 67150789 IC50 = 556 nM T61722 CGE76N 67218808 Ki = 86 nM T61722 C4CL2E 67218973 Ki = 2230 nM T61722 CJ1H6M 67219255 IC50 = 24 nM T61722 CV6UF7 67219271 IC50 = 4 nM T61722 CTNE42 67219428 IC50 = 147 nM T61722 C0WK1P 67242411 IC50 = 130 nM T61722 C2T0FW 67273087 IC50 = 20 nM T61722 CFUV51 67274014 IC50 = 7 nM T61722 CGNR25 67287864 IC50 = 22 nM T61722 C8IZ1A 67358288 IC50 = 145 nM T61722 CUG8B1 67494651 Ki = 4.9 nM T61722 C01UST 67494892 Ki = 2 nM T61722 C64FDJ 67496758 Ki = 750 nM T61722 C2BIX6 67496929 Ki = 16 nM T61722 CD4S8N 67497060 Ki = 96 nM T61722 CB80PW 67497062 Ki = 110 nM T61722 C9WQG5 67497152 Ki = 390 nM T61722 C75BRD 67497303 Ki = 490 nM T61722 CP9T0G 67497524 Ki = 280 nM T61722 CU0EX4 67606723 IC50 = 5000 nM T61722 CZIN41 67606737 IC50 = 1600 nM T61722 CVP16A 67606768 IC50 = 850 nM T61722 CSJL59 67606899 IC50 = 24 nM T61722 CVP0Z5 67607119 IC50 = 66 nM T61722 CZQK83 67607141 IC50 = 160 nM T61722 CMT76S 67607161 IC50 = 89 nM T61722 C0OHL8 67607174 IC50 = 5000 nM T61722 CG3NT9 67607179 IC50 = 7 nM T61722 C98MHU 67607200 IC50 = 81 nM T61722 CTH7J8 67607241 IC50 = 5000 nM T61722 CDX48U 67607248 IC50 = 490 nM T61722 C8HT0N 67607274 IC50 = 1400 nM T61722 C89JYX 67607503 IC50 = 2000 nM T61722 C1OA6C 67607812 IC50 = 5000 nM T61722 CP28AB 67608154 IC50 = 100 nM T61722 C7E4NZ 67609133 IC50 = 870 nM T61722 CO75NL 68011817 Ki = 35 nM T61722 C1WI5U 68349274 Ki = 18.3 nM T61722 CC93ZD 68349502 Ki = 1.6 nM T61722 CVM9Q1 68503758 IC50 = 275 nM T61722 CA15ND 68505312 IC50 = 23 nM T61722 C0US2T 68505327 IC50 = 4 nM T61722 CX8W7F 68508048 IC50 = 190 nM T61722 C9JDZ0 68509240 IC50 = 1590 nM T61722 C63FNH 69313615 IC50 = 2900 nM T61722 CP51CJ 69313717 IC50 = 72 nM T61722 C2OI8Z 69313931 IC50 = 1240 nM T61722 C4I3GV 69314007 IC50 = 9 nM T61722 CE85BW 69314646 IC50 = 980 nM T61722 C6VJ4M 69314659 IC50 = 150 nM T61722 C5UF0M 69314791 IC50 = 4410 nM T61722 CKU60M 69314812 IC50 = 2360 nM T61722 C57OGI 69314839 IC50 = 2200 nM T61722 C6GM3S 69315080 IC50 = 1400 nM T61722 COJ4Q1 69315206 IC50 = 2 nM T61722 CETR75 69315587 IC50 = 5 nM T61722 CJ5Z7T 69316129 IC50 = 15 nM T61722 C3JS8M 69316151 IC50 = 1.7 nM T61722 CH0P2Z 69316495 IC50 = 33 nM T61722 CIRN35 69316694 IC50 = 10 nM T61722 C7BCY2 69316753 IC50 = 41 nM T61722 CU9YH4 69316952 IC50 = 1360 nM T61722 CB04GT 69317123 IC50 = 5 nM T61722 C7N1VH 69317289 IC50 = 2690 nM T61722 C9HZD3 69317304 IC50 = 2 nM T61722 CDGE93 69318895 IC50 = 495 nM T61722 C45ZSM 69318939 IC50 = 1100 nM T61722 CDE59U 69319076 IC50 = 786 nM T61722 CJIF83 69319218 IC50 = 89 nM T61722 CD23LU 69319343 IC50 = 7690 nM T61722 CZS2G0 69319458 IC50 = 94 nM T61722 CFGB42 69319508 IC50 = 107 nM T61722 CHT8W2 69457082 IC50 = 520 nM T61722 CBK6R8 69465230 IC50 = 160 nM T61722 CAQ2K1 70681414 IC50 = 4 nM T61722 CAYQ23 70681415 IC50 = 10 nM T61722 C7JGK4 70681543 Ki = 631 nM T61722 CLGJ02 70681999 IC50 = 72 nM T61722 CIQF90 70682000 IC50 = 105 nM T61722 CQW5S4 70682001 IC50 = 810 nM T61722 CLW98J 70682002 IC50 = 10600 nM T61722 C1Z2JA 70682003 IC50 = 380 nM T61722 CY2TX8 70682004 IC50 = 470 nM T61722 CM7T9W 70683533 IC50 = 3.2 nM T61722 C3A4LS 70683534 IC50 = 18 nM T61722 CNJ92H 70683656 Ki = 492 nM T61722 C8F5SB 70683657 Ki = 591 nM T61722 CEB18O 70684120 IC50 = 1600 nM T61722 CUAV04 70685629 IC50 = 3.4 nM T61722 CS7I0V 70685804 Ki = 574 nM T61722 CTXI52 70685999 Ki = 4300 nM T61722 C14KHP 70686259 IC50 = 186 nM T61722 CCEM20 70686260 IC50 = 1200 nM T61722 CJ12SN 70686261 IC50 = 740 nM T61722 CTX51S 70687200 EC50 = 99 nM T61722 CUC4X0 70687356 IC50 = 11000 nM T61722 CVAX78 70687779 IC50 = 330 nM T61722 C57WTS 70687780 IC50 = 14 nM T61722 C17SDL 70687781 IC50 = 45 nM T61722 C57WBM 70687924 Ki = 563 nM T61722 C9WRA0 70688124 Ki = 8000 nM T61722 CVT87X 70688380 IC50 = 210 nM T61722 C12XDQ 70688381 IC50 = 370 nM T61722 C6TB1K 70689410 IC50 = 8 nM T61722 C6BFC9 70689411 IC50 = 15 nM T61722 CYO9K7 70689823 IC50 = 7.9 nM T61722 C3CR2K 70689824 IC50 = 3.2 nM T61722 CMZK24 70689956 Ki = 752 nM T61722 CCL56U 70689957 Ki = 520 nM T61722 CIU47N 70690398 IC50 = 370 nM T61722 C0DC1J 70691517 IC50 = 70 nM T61722 CP1YO8 70691973 IC50 = 4 nM T61722 C7QE0K 70691974 IC50 = 4.9 nM T61722 CPU36K 70691975 IC50 = 17 nM T61722 C0IWR2 70692435 IC50 = 7.4 nM T61722 C76WGV 70692569 IC50 > 10000 nM T61722 CM1SB9 70692570 IC50 = 580 nM T61722 CZ07KY 70692571 IC50 = 15 nM T61722 CTP4W6 70693611 IC50 = 7 nM T61722 C40EGX 70693612 IC50 = 30 nM T61722 CFC09Z 70694622 IC50 = 220 nM T61722 CN42UV 70695720 IC50 = 6 nM T61722 CAGV62 70695721 IC50 = 29 nM T61722 CE2KX9 70696139 IC50 = 83 nM T61722 C4WG2K 70696140 IC50 = 290 nM T61722 C73JLA 70696284 Ki = 623 nM T61722 C5ZPF2 70696285 Ki = 333 nM T61722 C3S6FN 70696448 Ki = 330 nM T61722 CY71SU 70696658 IC50 = 11400 nM T61722 CPFX95 70696659 IC50 = 220 nM T61722 CLE7P9 70696660 IC50 = 4 nM T61722 CD9LQ1 71118141 Ki = 3.4 nM T61722 COI5M1 71118253 Ki = 4 nM T61722 C7CI6X 71118509 Ki = 5 nM T61722 C7UTX6 71128570 Ki = 10 nM T61722 CB37RW 71128619 Ki = 9.4 nM T61722 CLVQ12 71128667 IC50 = 2.4 nM T61722 CTJ07K 71128670 Ki = 25 nM T61722 CTU38S 71135161 Ki = 3 nM T61722 C6PX5O 71139243 Ki = 32 nM T61722 C6C9ZD 71222485 IC50 = 10 nM T61722 CI5WE3 71222487 IC50 = 10 nM T61722 CWS2F0 71222492 IC50 = 4.7 nM T61722 CYQ17T 71222494 IC50 = 9 nM T61722 C13LBF 71222500 IC50 = 19 nM T61722 C5VNC8 71222501 IC50 = 82 nM T61722 C81XZD 71222503 IC50 = 1.4 nM T61722 CI0PB7 71222507 IC50 = 23 nM T61722 CM38YN 71222510 IC50 = 11 nM T61722 CUY54X 71222512 IC50 = 7 nM T61722 C3D9OG 71222513 IC50 = 15 nM T61722 CT7PK9 71222517 IC50 = 8 nM T61722 CIN24O 71222519 IC50 = 15 nM T61722 C4JB0K 71222531 IC50 = 5 nM T61722 C30PGM 71222534 IC50 = 127 nM T61722 CF1C4U 71222535 IC50 = 135 nM T61722 CNK9T5 71222559 IC50 = 15 nM T61722 CAD4C8 71222566 IC50 = 71 nM T61722 C1OB8N 71222570 IC50 = 23 nM T61722 CPYB97 71222574 IC50 = 108 nM T61722 C80FJW 71222598 IC50 = 19 nM T61722 C4DSV1 71222679 IC50 = 49 nM T61722 CCO6V5 71223324 IC50 = 37 nM T61722 C5ED7W 71223325 IC50 = 6.3 nM T61722 CR6A7Z 71223330 IC50 = 19 nM T61722 C1EM7Z 71223479 IC50 = 9 nM T61722 C2UO8S 71223491 IC50 = 33 nM T61722 C47AGQ 71223494 IC50 = 37 nM T61722 CCV21X 71223526 IC50 = 14 nM T61722 C0LP3T 71223554 IC50 = 2 nM T61722 C64HKL 71223571 IC50 = 11 nM T61722 CBZ4O7 71223583 IC50 = 4.3 nM T61722 C0TDZ9 71225451 IC50 = 2 nM T61722 CSF90B 71225486 IC50 = 5 nM T61722 C52KPS 71225493 IC50 = 2 nM T61722 C7WVM9 71225497 IC50 = 1 nM T61722 CQNX28 71225530 IC50 = 5 nM T61722 CKB2W3 71225606 IC50 = 4 nM T61722 C3Q6OL 71225631 IC50 = 10 nM T61722 C1VR6C 71225636 IC50 = 4 nM T61722 CS97ML 71225655 IC50 = 16 nM T61722 C3OTB0 71225700 IC50 = 1800 nM T61722 C50RED 71225703 IC50 = 4.7 nM T61722 CC9RW4 71225712 IC50 = 28 nM T61722 CWB2K6 71225716 IC50 = 8.5 nM T61722 CG91OC 71225722 IC50 = 5.8 nM T61722 C52GTH 71225735 IC50 = 29 nM T61722 CSN7E8 71225753 IC50 = 163 nM T61722 C6SOB3 71225773 IC50 = 3 nM T61722 C9KQT4 71225800 IC50 = 6 nM T61722 CP9GU5 71225801 IC50 = 97 nM T61722 C3R9AS 71225803 IC50 = 5 nM T61722 CZ5X9I 71225804 IC50 = 3 nM T61722 C7YJB8 71225823 IC50 = 3 nM T61722 CV3BL1 71225896 IC50 = 6 nM T61722 CZ68QJ 71225916 IC50 = 7.7 nM T61722 C6AL1H 71225932 IC50 = 150 nM T61722 CC0B5G 71225937 IC50 = 2 nM T61722 C8BKO4 71225985 IC50 = 8 nM T61722 CDAQ09 71226066 IC50 = 10 nM T61722 CD36LO 71226099 IC50 = 4.2 nM T61722 C79MAS 71226106 IC50 = 64 nM T61722 CTP1E2 71226159 IC50 = 1000 nM T61722 C1TGK5 71226404 IC50 = 7 nM T61722 C95YNA 71226725 IC50 = 2600 nM T61722 C95NPO 71226942 IC50 = 119 nM T61722 CQXS19 71227039 IC50 = 16 nM T61722 CM12EU 71450296 IC50 = 18 nM T61722 C7T1LK 71459331 IC50 = 2 nM T61722 CF7A3H 71459332 IC50 = 34 nM T61722 C05UTH 71463001 IC50 > 1000 nM T61722 C0GW3I 71470140 IC50 = 240 nM T61722 CHC3J0 71470142 IC50 = 6 nM T61722 CT17XU 71470226 IC50 = 3.6 nM T61722 CD3L0A 71470229 IC50 = 480 nM T61722 C5G9DO 71470300 IC50 = 810 nM T61722 C6HWS1 71470301 IC50 = 4 nM T61722 CR9EA0 71470382 IC50 = 5 nM T61722 CJ7K6W 71470383 IC50 = 5 nM T61722 CZH56E 71470386 IC50 = 4.9 nM T61722 C47KLT 71470472 IC50 = 2.2 nM T61722 CB50YZ 71470556 IC50 = 32 nM T61722 CMJA71 71470732 IC50 = 3 nM T61722 C9BQ0A 71470733 IC50 = 28 nM T61722 CG53LJ 71470848 IC50 = 3.6 nM T61722 C1X8ZT 71470938 IC50 = 3.3 nM T61722 CM9V6Y 71470939 IC50 = 7 nM T61722 C7KS9U 71470941 IC50 = 11 nM T61722 C51WTF 71470942 IC50 = 19 nM T61722 C6ZO3R 71470943 IC50 = 4 nM T61722 COD6P9 71471033 IC50 = 3 nM T61722 CRV58Y 71471034 IC50 = 13 nM T61722 C8F5DU 71471035 IC50 = 6.2 nM T61722 CCYN97 71471137 IC50 = 900 nM T61722 C3UQ0B 71471138 IC50 = 3.9 nM T61722 CV8I9B 71471139 IC50 = 8.5 nM T61722 CWM3P2 71471140 IC50 = 6.6 nM T61722 CQX1Z2 71471141 IC50 = 3.6 nM T61722 CGJX89 71471249 IC50 = 430 nM T61722 CBL6T2 71471250 IC50 = 91 nM T61722 C9PN3X 71471252 IC50 = 20 nM T61722 C89QZE 71471349 IC50 = 10 nM T61722 C6FBW9 71471350 IC50 = 550 nM T61722 C50WAT 71471351 IC50 = 4500 nM T61722 CD06QJ 71471352 IC50 = 12 nM T61722 CY8T5B 71471354 IC50 = 1.5 nM T61722 C91UTY 71471464 IC50 = 170 nM T61722 C0QCW9 71471465 IC50 = 3.7 nM T61722 CKA1U8 71471467 IC50 = 28 nM T61722 C3M8NK 71471469 IC50 = 530 nM T61722 CVFH19 71471569 IC50 = 26 nM T61722 C3XA5H 71471571 IC50 = 120 nM T61722 CY5D1U 71471572 IC50 = 3.9 nM T61722 CS5ZG0 71471574 IC50 = 9 nM T61722 CDF70S 71476538 IC50 = 0.9 nM T61722 C5Y3NV 71476981 IC50 = 1.7 nM T61722 CVD51W 71482237 IC50 = 23 nM T61722 CJE9N4 71482495 IC50 = 54 nM T61722 CS27QD 71482643 IC50 = 18 nM T61722 C9YHK3 71482644 IC50 = 5.9 nM T61722 CTA8J6 71482786 IC50 = 15 nM T61722 CHM3C8 71482787 IC50 = 6 nM T61722 CA5ZR0 71483542 IC50 = 40 nM T61722 CB23KI 71552007 IC50 = 5900 nM T61722 C4CR2L 71552008 IC50 = 2600 nM T61722 C8PWX0 71552009 IC50 = 510 nM T61722 CAP4L3 71552010 IC50 = 560 nM T61722 C5RM9E 71552087 IC50 = 4400 nM T61722 CXS3M0 71552088 IC50 = 10 nM T61722 CK7WR2 71552089 IC50 = 10 nM T61722 CV7TG4 71552090 IC50 = 45 nM T61722 C1IE4J 71552158 IC50 = 100 nM T61722 C8TQI1 71552159 IC50 = 5 nM T61722 CX4KL3 71552160 IC50 = 7 nM T61722 CIEX50 71552161 IC50 = 290 nM T61722 C5XW7L 71552162 IC50 = 50 nM T61722 CMP7L3 71552163 IC50 = 10 nM T61722 C0Z1DT 71552164 IC50 = 7 nM T61722 CX2IN5 71552246 IC50 = 690 nM T61722 C0P4OW 71552247 IC50 = 140 nM T61722 CC2A4K 71552667 IC50 = 490 nM T61722 CPX2U5 71624847 IC50 = 230 nM T61722 C49SMN 71624848 IC50 > 5000 nM T61722 CBX43D 71624850 IC50 = 36 nM T61722 CN9C4G 71624851 IC50 = 2900 nM T61722 C27DEO 71624966 IC50 = 4 nM T61722 CA1EN7 71624967 IC50 = 46 nM T61722 CFJC91 71624968 IC50 = 1900 nM T61722 C19WPA 71624969 IC50 = 290 nM T61722 CGX1Y7 71625096 IC50 = 1100 nM T61722 CLU9T6 71625097 IC50 = 5000 nM T61722 CD62SQ 71733817 IC50 = 35 nM T61722 C8XJ0I 71733818 IC50 = 180 nM T61722 CXC78L 71733909 IC50 = 20 nM T61722 C7B5XE 71733910 IC50 = 70 nM T61722 CQ21ZD 71733911 IC50 = 50 nM T61722 CZG0S2 71733912 IC50 = 10 nM T61722 CK37JI 72736342 IC50 = 220 nM T61722 C4BQJ7 72736343 IC50 = 21 nM T61722 C01PVO 72736344 IC50 = 400 nM T61722 CW8F7N 72736517 IC50 = 350 nM T61722 CZ7B5D 72736518 IC50 = 7.4 nM T61722 CK3G6N 72736699 IC50 = 322 nM T61722 CXVT85 72736700 IC50 = 67 nM T61722 C9T5DA 72736853 IC50 = 5.2 nM T61722 CR58HL 72736854 IC50 = 8.7 nM T61722 CJ1G8C 72736855 IC50 = 7.8 nM T61722 CP0TC3 72737017 IC50 = 6.2 nM T61722 CPH2N7 72737018 IC50 = 14 nM T61722 CUQ3E6 72737019 IC50 = 14 nM T61722 CKF7W9 72737020 IC50 = 15 nM T61722 CS9HB3 72737190 IC50 = 9.9 nM T61722 C5JCZ7 72737191 IC50 = 8.2 nM T61722 CX9Z8F 72737383 IC50 = 3.7 nM T61722 CLI58Z 72737384 IC50 = 85 nM T61722 C0G2IM 73347358 IC50 = 1600 nM T61722 C4UZR9 73348867 IC50 = 310 nM T61722 CC5AL2 76310043 IC50 = 2000 nM T61722 CDB2L0 76310044 IC50 = 160 nM T61722 CVE2Y6 76310045 IC50 = 110 nM T61722 CA7RB5 76310046 IC50 = 4000 nM T61722 C89JPW 76310047 IC50 = 50 nM T61722 C4QWV8 76310885 Ki = 41.7 nM T61722 CU3XV9 76310898 Ki = 2.5 nM T61722 C73AST 76310899 Ki = 1.1 nM T61722 C9X2AC 76313695 IC50 = 50 nM T61722 CVY95B 76313754 IC50 = 5000 nM T61722 CE94AX 76313755 IC50 = 520 nM T61722 CL7B1W 76313756 IC50 = 4 nM T61722 CTO8Z3 76313757 IC50 = 110 nM T61722 CF38TZ 76313758 IC50 = 50 nM T61722 CB68VZ 76314517 Ki = 1.9 nM T61722 C5XT6K 76314537 Ki = 19.6 nM T61722 C5TRD4 76314538 Ki = 5.6 nM T61722 C3PSV5 76314539 Ki = 1.8 nM T61722 C37MNV 76314540 Ki = 10.5 nM T61722 CS86VL 76317265 IC50 = 220 nM T61722 CI0K2W 76317266 IC50 = 200 nM T61722 CC2X9M 76317267 IC50 = 380 nM T61722 CF3WP1 76317268 IC50 = 200 nM T61722 CF2EA8 76317269 IC50 = 470 nM T61722 CV7OJ4 76318094 Ki = 3.7 nM T61722 CP8YK5 76318114 Ki = 3 nM T61722 CV3E6G 76320915 IC50 = 48 nM T61722 CNF6M4 76320969 IC50 = 300 nM T61722 C4LDJ8 76320970 IC50 = 2300 nM T61722 CC1O9U 76324644 IC50 = 5000 nM T61722 CSGR40 76324645 IC50 = 720 nM T61722 C95BSK 76325442 Ki = 2.6 nM T61722 C9O8KW 76325443 Ki = 6 nM T61722 CG03LZ 76325444 Ki = 22.3 nM T61722 CGH5C0 76328208 IC50 = 87 nM T61722 C6BV9D 76328209 IC50 = 70 nM T61722 CYO1Z6 76328210 IC50 = 1100 nM T61722 C4RBP5 76328211 IC50 = 450 nM T61722 CP5XO2 76328212 IC50 = 110 nM T61722 CVR68K 76328965 Ki = 7.4 nM T61722 C7TWH4 76328986 Ki = 13.7 nM T61722 CM3A0Y 76331881 IC50 = 400 nM T61722 CYG9N4 76331882 IC50 = 60 nM T61722 C7V4HI 76331883 IC50 = 230 nM T61722 COB4M1 76331884 IC50 = 5000 nM T61722 C2SK8J 76331886 IC50 = 450 nM T61722 CQ7LK2 76332661 Ki = 1.8 nM T61722 CC62DQ 76335451 IC50 = 440 nM T61722 COYJ34 76335452 IC50 = 2500 nM T61722 CR71KA 76335453 IC50 = 270 nM T61722 CI68LE 76335454 IC50 = 1600 nM T61722 CA5XS9 76335455 IC50 = 70 nM T61722 C64TPS 76336263 Ki = 3.7 nM T61722 C3VB0G 76336264 Ki = 4.1 nM T61722 CZF5R9 76336265 Ki = 3.4 nM T61722 CQYR65 76336266 Ki = 24.9 nM T61722 CT60NR 76336267 Ki = 2 nM T61722 C92DQZ 87314562 IC50 = 14 nM T61722 COW62K 90094257 Ki = 0.23 nM T61722 C1U3FE 90094966 Ki = 4920 nM T61722 CLFX12 90095044 Ki = 14 nM T61722 CWHO10 90095087 Ki = 0.4 nM T61722 CW76HC 90095106 Ki = 9.2 nM T61722 C43KBQ 90095410 Ki = 24 nM T61722 CA9VG0 90095663 Ki = 49 nM T61722 C6U8SR 90095975 Ki = 21 nM T61722 CF4WL8 90096261 Ki = 1.31 nM T61722 CK2V7U 90096263 Ki = 15 nM T61722 CGBQ38 90479860 IC50 = 31 nM T61722 CKD3U1 90644206 IC50 = 57 nM T61722 CGP87O 90644207 IC50 = 56 nM T61722 CK13SY 90644208 IC50 = 32 nM T61722 CJNR26 90644209 IC50 = 32 nM T61722 C0JVX4 90655032 IC50 = 52 nM T61722 CL1D7B 90655033 IC50 > 2000 nM T61722 C7E0TD 90655034 IC50 > 2000 nM T61722 CN98XT 90655035 IC50 > 2000 nM T61722 CR9VW6 90655036 IC50 > 2000 nM T61722 C96YLX 90655037 IC50 = 689 nM T61722 C8P5QX 90655038 IC50 > 2000 nM T61722 CC8SK0 90655039 IC50 > 2000 nM T61722 C84VJT 118558137 Ki = 13 nM T61722 C5KH9L 118558148 Ki = 8.5 nM T61722 CE67GI 118558154 Ki = 19 nM T61722 C85UXH 118715115 IC50 = 240 nM T61722 C18DAH 118715116 IC50 = 800 nM T61722 C6THR1 118715117 IC50 = 16 nM T61722 CKVA04 118715118 IC50 = 48 nM T61722 C7H1PL 118715119 IC50 = 48 nM T61722 C89NFI 118715120 IC50 = 398 nM T61722 C16PZI 118715121 IC50 = 159 nM T61722 C9BS3H 118715122 IC50 = 247 nM T61722 CE31JP 118715123 IC50 = 123 nM T61722 COWU53 118715124 IC50 = 262 nM T61722 CIC0V4 118715125 IC50 = 8 nM T61722 CJEN92 118715174 IC50 = 4 nM T61722 C0ABO8 118715176 IC50 = 27 nM T61722 CCY19P 118715180 IC50 = 51 nM T61722 COX6U0 118715181 IC50 = 580 nM T61722 CTY95E 118715182 IC50 = 250 nM T61722 C5J6HW 118715183 IC50 = 30 nM T61722 C3U2IO 118715184 IC50 = 1400 nM T61722 C5UM3H 118715185 IC50 = 170 nM T61722 CMC5Q8 118715186 IC50 = 7 nM T61722 CNP4R9 118715187 IC50 = 5 nM T61722 CDE6U0 118715188 IC50 = 20 nM T61722 CQL41Z 118715189 IC50 = 7 nM T61722 C7VLX9 118715190 IC50 = 4 nM T61722 CJF15Z 118715191 IC50 = 6 nM T61722 C4XD0U 118716858 IC50 = 11 nM T61722 CZYH52 118716859 IC50 = 4 nM T61722 C5LS6K 118716860 IC50 = 4 nM T61722 CHEY81 118716861 IC50 = 14 nM T61722 CAQK39 127029906 IC50 = 104 nM T61722 C5DBA3 127029907 IC50 = 2 nM T61722 C4OSF7 127030244 IC50 = 1600 nM T61722 CM5E4R 127030245 IC50 = 3000 nM T61722 CT0PV9 127031167 IC50 = 2400 nM T61722 CE4DH9 127031169 IC50 = 8 nM T61722 C2G5HL 127031170 IC50 = 10000 nM T61722 CQ26EX 127031171 IC50 = 860 nM T61722 CVJ5L2 127032055 IC50 = 18 nM T61722 C5WO4N 127032356 IC50 = 970 nM T61722 C4BPL3 127032357 IC50 = 10000 nM T61722 CP51ET 127033310 IC50 = 12 nM T61722 CK1G5P 127033311 IC50 = 47 nM T61722 C15HZP 127033547 IC50 = 2 nM T61722 C4FJO8 127033599 IC50 = 14 nM T61722 C2C5JT 127033600 IC50 = 5 nM T61722 CQ27PR 127033601 IC50 = 4 nM T61722 CI9AK0 127034111 IC50 = 65 nM T61722 CUM17V 137637879 Ki = 72 nM T61722 C25HXF 137643575 IC50 = 6 nM T61722 C0VRX4 137651001 Ki = 1335 nM T61722 C7Z4JW 137656723 Ki = 735 nM T61722 CDMF42 145963927 Ki = 9 nM T61722 CFZC50 145964169 Ki = 7800 nM T61722 CP93WL 145964478 Ki = 110 nM T61722 CRZL87 145964698 Ki = 7.8 nM T61722 C3XI4Q 145964823 Ki = 98 nM T61722 C1VK6G 145965291 IC50 = 0.8 nM T61722 CB8H1L 145965334 Ki = 26 nM T61722 CQW53X 145965434 Ki = 56 nM T61722 C4XOC5 145965717 Ki = 16 nM T61722 CKM0Q8 145965834 Ki = 703 nM T61722 CWN82U 145966000 Ki = 38 nM T61722 CD9Y5A 145966022 Ki = 2.3 nM T61722 CJ93HP 145966539 Ki = 43 nM T61722 CV4N2L 145966642 Ki = 7.3 nM T61722 CBU14Z 145967014 Ki = 13 nM T61722 CUI90K 145967050 Ki = 26 nM T61722 CV3H9X 145967484 Ki = 6 nM T61722 CW6XM1 145967527 Ki = 22 nM T61722 C4YTR2 145968674 Ki = 3.5 nM T61722 CS4F5A 145970055 Ki = 1490 nM T61722 C8F7HJ 145970970 Ki = 8.1 nM T61722 C2GSZ1 145971410 Ki = 11 nM T61722 C3MZF6 145971559 Ki = 660 nM T61722 CEW7B4 145972084 Ki = 50 nM T61722 C41OSC 145972617 Ki = 510 nM T61722 C91URI 145973046 Ki = 12 nM T61722 CR9FG0 145974144 Ki = 5 nM T61722 CR76AV 145974214 Ki = 14 nM T61722 CMS2N4 145974264 Ki = 840 nM T61722 CZU07L 145974722 Ki = 31 nM T61722 CJBZ64 145975085 Ki = 28 nM T61722 CHNP49 145975308 Ki = 7 nM T61722 C0K5QT 145975859 Ki = 82 nM T61722 C0O7IR 145975984 Ki = 64 nM T61722 C4M0XE 145976613 Ki = 300 nM T61722 CA8G7P 145976943 EC50 = 12 nM T61722 CZ71CN 145977428 Ki = 12 nM T61722 CV4M5B 145978653 Ki = 14 nM T61722 C8ZA9D 145978688 Ki = 8.6 nM T61722 C75YEA 145978844 Ki = 35 nM T61722 D00GUE 46230226 IC50 = 370 nM T61722 D01AFV 11500603 Ki = 83 nM T61722 D02MXT 24952929 Ki > 21000 nM T61722 D05GWV 11586961 Ki = 230 nM T61722 D05HPB 11587023 Ki = 782 nM T61722 D07GCA 11514705 Ki = 59 nM T61722 D08CLB 346737 Ki = 311 nM T61722 D08KZJ 11384493 Ki = 0.6 nM T61722 D09ZSV 968879 IC50 = 481 nM T61722 D0C0FU 43091550 Ki = 3280 nM T61722 D0E0HT 248828 Ki = 5130 nM T61722 D0E3WT 2763923 IC50 = 870 nM T61722 D0H2SL 719761 IC50 = 61 nM T61722 D0I8MN 44441193 Ki = 150 nM T61722 D0J2PW 46533 IC50 = 1970 nM T61722 D0J5OX 16775011 Ki = 799 nM T61722 D0M2DJ 19261363 IC50 = 4520 nM T61722 D0QE3V 44403763 Ki = 0.8 nM T61722 D0QH5C 230826 Ki = 154 nM T61722 D0R1KE 894151 IC50 = 6870 nM T61722 D0S0BK 44441192 Ki = 353 nM T61722 D0U3LA 44417452 IC50 = 437 nM T61722 D0U5PC 43169594 Ki = 1990 nM T61722 D0Y4UG 44441190 Ki = 446 nM T62390 CD27TG 5311191 IC50 = 1000 nM T62390 CRQN68 10333842 IC50 = 42000 nM T62390 CPNA96 13922235 IC50 = 87000 nM T62390 D06LQH 167715 IC50 = 300 nM T62390 D0CI3A 439744 IC50 = 720 nM T51597 D03OIW 3830 IC50 > 1000000 nM T51597 D0E1SW 1986 IC50 > 1000000 nM T51597 CVH86L 10661 IC50 > 2500000 nM T51597 CN35IZ 119339 IC50 = 40 nM T51597 C4YJ5D 205045 IC50 = 13000 nM T51597 CTNY78 449124 IC50 = 4500 nM T51597 C3C8PN 823788 IC50 = 40000 nM T51597 CC57PQ 1790942 IC50 = 100000 nM T51597 CF6SI1 2730721 IC50 = 80000 nM T51597 C0TFQ9 2813100 IC50 = 700 nM T51597 CF8Y4N 2814578 IC50 = 30000 nM T51597 CBZ7P2 2928097 Ki = 3960 nM T51597 CSP68E 3040782 IC50 = 22000 nM T51597 CERF41 3151315 Ki = 9720 nM T51597 C57FID 6522754 IC50 = 4000 nM T51597 CL4GK5 13686033 IC50 = 210 nM T51597 C81GKF 15019055 IC50 = 15000 nM T51597 C6VFC9 16785637 IC50 = 101700 nM T51597 CX83UG 118165178 IC50 > 100000 nM T51597 CWX3Z7 118165190 IC50 > 100000 nM T51597 C3S5OA 118165200 IC50 = 73 nM T51597 C95RGM 118165205 IC50 > 100000 nM T51597 C3Y0TE 118165222 IC50 > 3325 nM T51597 CE9Z3K 118165243 IC50 = 5.4 nM T51597 C2VZW7 118165257 IC50 = 182 nM T51597 CIJN30 118165260 IC50 = 1545 nM T51597 CA8YG6 118165270 IC50 > 100000 nM T51597 C84VSY 118165287 IC50 = 8.7 nM T51597 C6X5HK 118165290 IC50 = 3.4 nM T51597 CNFT52 118165293 IC50 = 18450 nM T51597 CB59GF 118165313 IC50 = 348 nM T51597 CFIV09 118165354 IC50 = 660 nM T51597 CZ8RQ9 118165413 IC50 = 970 nM T51597 C3F6XG 118165440 Ki = 13.5 nM T51597 CWI08V 118165445 IC50 = 13200 nM T51597 CA9E0U 118165472 IC50 = 1111 nM T51597 CDAC50 118165497 IC50 = 111 nM T51597 CWP90I 118165555 IC50 > 100000 nM T51597 CM6JI8 118165621 IC50 = 134 nM T51597 C8V1IU 118165625 IC50 = 4137 nM T51597 CNPW85 118165709 IC50 = 3.5 nM T51597 CAZ25P 118165748 IC50 = 2025 nM T51597 C65DLT 118165752 IC50 > 100000 nM T51597 CA9UQ1 118165756 IC50 = 8.7 nM T51597 CATZ25 118165760 IC50 = 12250 nM T51597 CN4O5K 118165763 IC50 = 98 nM T51597 CR5HV8 121410292 IC50 = 28 nM T51597 CVE96K 121410294 IC50 = 163 nM T51597 CK9G7V 121410328 IC50 = 690 nM T51597 CQ3KL4 121410329 IC50 = 425 nM T51597 CBN62U 121410340 IC50 = 1040 nM T51597 CNF06J 121410352 IC50 = 37 nM T51597 CR70JL 126641909 IC50 = 23 nM T51597 CT7M6Q 126641926 IC50 = 39 nM T51597 CLG67Z 126641948 IC50 = 22 nM T51597 CVAC39 126641974 IC50 = 395 nM T51597 C1ZTB7 126641995 IC50 = 26 nM T51597 CA81IH 126642266 IC50 = 19 nM T51597 CNJL38 126642277 IC50 = 73 nM T51597 CIW02N 126642282 IC50 = 50 nM T51597 CM65EN 135552113 IC50 = 100000 nM T51597 CO09EN 155514507 IC50 = 83 nM T51597 CGWL21 155515495 IC50 = 1350 nM T51597 CPZ1J2 155515757 IC50 = 135 nM T51597 CVS35D 155518925 IC50 = 40 nM T51597 CS0ER5 155528109 IC50 = 185 nM T51597 C2WPD6 155530588 IC50 = 68 nM T51597 CYH2Z6 155530878 IC50 = 135 nM T51597 CGKM58 155542422 IC50 = 103 nM T51597 CN9LP5 155551221 IC50 = 21 nM T51597 CGV1M3 155552611 IC50 = 28 nM T51597 CM5VI1 155561970 IC50 = 5950 nM T99041 D02EYG 10096344 IC50 = 0.1 nM T99041 D04AIT 5280445 IC50 = 120 nM T99041 D07MGA 72281 IC50 = 280 nM T99041 D0D7LA 4091 IC50 = 29000 nM T99041 D0K8KX 5280343 IC50 = 32730 nM T99041 D0K9MY 11243969 Ki = 0.6 nM T99041 D0L3DK 6918537 Ki = 3 nM T99041 D0N5HJ 5462501 IC50 > 100000 nM T99041 D0NI0C 21704 IC50 = 62 nM T99041 D0NJ5H 11450633 IC50 = 2.7 nM T99041 D0RA5Q 72172 IC50 > 100 ug.mL-1 T99041 D0T8XB 44513473 IC50 = 3.8 nM T99041 D0U2JP 4369359 IC50 = 3.5 nM T99041 D0Y7LD 222284 IC50 = 28840 nM T99041 D04XIO 11253490 IC50 = 23 nM T99041 D05LPW 25022354 IC50 = 0.9 nM T99041 D07EPV 11949652 IC50 = 0.37 nM T99041 D07HZG 11516136 IC50 = 11.3 nM T99041 D0FQ2U 6918572 Ki = 0.18 nM T99041 D0L4FS 5280961 IC50 = 480 nM T99041 D0M3XR 46209133 Ki = 0.8 nM T99041 D0N6SO 15983988 IC50 = 4 nM T99041 D0R9HL 11077541 IC50 = 3.5 nM T99041 D0R9YR 64971 IC50 = 55820 nM T99041 D0U2BH 65064 IC50 = 10210 nM T99041 D0U3EP 445154 IC50 = 0.6 nM T99041 D02LNB 22387295 IC50 = 12 nM T99041 D04MAZ 71731606 IC50 = 0.4 nM T99041 D05FMP 66561557 IC50 > 100000 nM T99041 D07JHU 71667377 IC50 > 100000 nM T99041 D0C6NX 73356493 IC50 > 100000 nM T99041 D0K2ZQ 57378228 IC50 = 0.42 nM T99041 D0QX2U 71667229 IC50 > 100000 nM T99041 D00FYF 9796290 IC50 = 22 nM T99041 D01XGX 178060 IC50 > 100000 nM T99041 D08PUW 64982 IC50 = 225000 nM T99041 D0A1NU 16049769 Ki = 1 nM T99041 D0F3TI 11673176 Ki = 1.8 nM T99041 D0Q4YP 11996845 IC50 = 5.3 nM T99041 D0T2IQ 443600 IC50 > 100 ug.mL-1 T99041 CR40US 18844 IC50 = 7 nM T99041 CT2EY7 56877 IC50 > 100000 nM T99041 CL1Y4H 68247 IC50 = 1410 nM T99041 CBP13T 69512 IC50 = 1410 nM T99041 C0V9WL 73324 IC50 > 100 ug.mL-1 T99041 CHAI28 83489 IC50 = 10360 nM T99041 C8EQ1Z 92855 IC50 = 35600 nM T99041 CP1JX4 124031 IC50 = 23.4 ug.mL-1 T99041 C15AMW 158341 IC50 = 14130 nM T99041 CB9Q1L 168182 IC50 = 65690 nM T99041 C6JM7L 182750 IC50 > 100 ug.mL-1 T99041 CV0J8H 182751 IC50 > 100 ug.mL-1 T99041 CGT6C5 276114 IC50 > 100 ug.mL-1 T99041 C7HME8 439246 IC50 = 240 nM T99041 CT2S6P 441667 IC50 = 420 nM T99041 CPKO72 448436 IC50 = 0.1 nM T99041 CP3EL4 454740 IC50 = 3350 nM T99041 C0GD3A 454742 IC50 = 890 nM T99041 C0TYO2 477693 IC50 = 19.8 ug.mL-1 T99041 C7G3CT 477696 IC50 > 100 ug.mL-1 T99041 C8P2LC 485077 IC50 = 56230 nM T99041 CG3C4U 489605 IC50 = 25000 nM T99041 CSJ38Y 679638 IC50 = 3900 nM T99041 CPEY84 688304 IC50 > 100000 nM T99041 C4TRL6 721814 IC50 > 337500 nM T99041 CO3KZ2 741570 IC50 > 100 ug.mL-1 T99041 C18XUS 978607 IC50 = 2800 nM T99041 C0L7TD 1235479 IC50 = 81 ug.mL-1 T99041 C2HQJ7 2302144 IC50 > 100 ug.mL-1 T99041 C30WIA 2750782 IC50 > 100000 nM T99041 CJW0G1 2854000 IC50 = 4000 nM T99041 CT2CQ8 3021908 IC50 = 21000 nM T99041 CX08LH 3081017 IC50 > 100000 nM T99041 CAZ25S 3318661 IC50 > 1000000 nM T99041 CQ0G4F 5281406 IC50 = 87100 nM T99041 C1DW0R 5316300 IC50 = 38430 nM T99041 CAU3O8 5317238 IC50 = 87720 nM T99041 CFB0N1 5318591 IC50 = 26920 nM T99041 CL6J0E 5320287 IC50 = 41690 nM T99041 CQP43H 5360349 IC50 = 5 nM T99041 CS5BG1 5494385 IC50 = 23 nM T99041 CDG53K 5494422 IC50 = 90 nM T99041 CT0E7G 6293081 IC50 = 33110 nM T99041 CE98OF 6451150 IC50 = 21.88 nM T99041 CPUF51 6918418 IC50 = 5700 nM T99041 C4RE5F 7020797 IC50 = 21000 nM T99041 C48BSO 7614279 IC50 = 26100 nM T99041 C37RIP 9655981 IC50 = 3440 nM T99041 C14VRG 9794073 IC50 = 3900 nM T99041 CQT36A 9794235 IC50 = 1700 nM T99041 CXEQ40 9795464 IC50 = 64 nM T99041 CMVO26 9795469 IC50 = 21 nM T99041 CBG8M2 9796291 IC50 = 1170 nM T99041 CSA6V9 9796352 Ki = 218 nM T99041 C7KR1T 9799867 IC50 = 4 nM T99041 CNJ0Z3 9800721 Ki = 2 nM T99041 C75RIB 9801978 IC50 = 7 nM T99041 C5F7DH 9815545 IC50 = 2 nM T99041 CUNB40 9817010 IC50 = 247000 nM T99041 C1I5JZ 9819537 IC50 = 298 nM T99041 CDP16K 9821063 IC50 = 17000 nM T99041 C8CR0Z 9821205 IC50 = 0.13 nM T99041 CKR9Y5 9823963 IC50 = 13 nM T99041 C8EK7G 9835053 IC50 = 3700 nM T99041 CW5EZ7 9835382 IC50 = 1600 nM T99041 CDY12G 9835472 IC50 = 3100 nM T99041 CV87XC 9835734 Ki = 154 nM T99041 CAHB35 9836210 IC50 = 922 nM T99041 CU2B0F 9838664 IC50 = 110 nM T99041 C62DNH 9843297 IC50 = 27 nM T99041 CUD46C 9855673 IC50 = 188000 nM T99041 CO2YQ4 9858442 IC50 = 69 nM T99041 C8XO1Z 9859008 Ki = 18 nM T99041 CNYI42 9859384 IC50 = 0.6 nM T99041 C2DMP6 9861924 IC50 > 100 ug.mL-1 T99041 CK0BS5 9864687 IC50 = 36 nM T99041 C5CZ6J 9865563 Ki = 53 nM T99041 CF3I8A 9865779 IC50 = 4.6 nM T99041 CR9AW7 9870934 IC50 = 23 nM T99041 CQN2L1 9882325 IC50 = 63 nM T99041 CZUQ34 9883487 IC50 = 460 nM T99041 C2TV9M 9884543 IC50 = 0.064 nM T99041 CBI2C9 9885607 IC50 = 82 nM T99041 CFMG63 9886974 IC50 = 12 ug.mL-1 T99041 CBW37X 9903629 IC50 = 466 nM T99041 C4T1CX 9904675 IC50 = 491 nM T99041 CU0I4K 9907074 IC50 = 270 nM T99041 CMGX12 9920733 IC50 = 23100 nM T99041 C4EC8A 9924995 IC50 = 610 nM T99041 C1S5VM 9927481 IC50 = 436 nM T99041 C6T0RU 9928326 IC50 = 360 nM T99041 C8Y5UK 9939534 IC50 = 23 nM T99041 CFH1V2 9942336 IC50 > 1000000 nM T99041 C28XTC 9942425 Ki = 2000 nM T99041 CZ1S9O 9942554 IC50 = 0.3 nM T99041 CZMT26 9947730 IC50 = 166 nM T99041 C2KW8I 9951445 IC50 = 1.8 nM T99041 CLR78W 9952894 IC50 = 88 nM T99041 CQ8J7T 9953181 IC50 = 59 nM T99041 C8OX9T 9964212 IC50 = 50400 nM T99041 C8THS1 9970277 IC50 = 64000 nM T99041 C1A3YN 9972358 IC50 = 2300 nM T99041 CH39FT 9973732 IC50 = 2000 nM T99041 C9EZ1X 9978478 IC50 = 2.2 nM T99041 CT6XQ2 9983092 IC50 = 1.4 nM T99041 C18ZXU 9990413 IC50 > 1000000 nM T99041 C1NB0Q 9992723 Ki = 79 nM T99041 C5Q6BJ 9995375 IC50 > 100 ug.mL-1 T99041 C17BCF 10003476 IC50 = 1 nM T99041 CN8XI3 10006926 IC50 = 1 nM T99041 CVG9I2 10012350 IC50 > 1000000 nM T99041 C7IB1W 10014222 Ki = 8 nM T99041 C4KT7I 10014539 IC50 > 1000000 nM T99041 CQ7G2R 10018887 IC50 = 1100 nM T99041 CV85MG 10019118 IC50 = 196000 nM T99041 CN0T5A 10019492 IC50 = 7400 nM T99041 C78NMY 10026124 IC50 = 234 nM T99041 CWQ21K 10038196 Ki = 96 nM T99041 CSZ75E 10046311 IC50 = 71 nM T99041 CRG1N0 10058240 IC50 >> 1000000 nM T99041 CYMG54 10058520 Ki = 210 nM T99041 C64ZDU 10059633 IC50 = 545000 nM T99041 CYH3C6 10061400 IC50 > 100 ug.mL-1 T99041 CV7SK8 10064801 IC50 = 57800 nM T99041 CI1Q6X 10081481 IC50 > 500000 nM T99041 CHC82B 10083376 IC50 > 1000000 nM T99041 CSHQ57 10084828 IC50 > 1000000 nM T99041 CB9J1F 10086451 IC50 = 16 nM T99041 C06KTL 10087724 IC50 > 1000000 nM T99041 C97FIB 10087948 IC50 = 245 nM T99041 C83ZDL 10096130 IC50 = 22 nM T99041 C8P3UC 10106636 Ki = 24 nM T99041 C5U0ON 10107122 IC50 = 3.3 nM T99041 C3K2MO 10109454 IC50 = 0.18 nM T99041 C7A3ZJ 10111068 Ki = 79 nM T99041 CKP5D7 10111288 IC50 = 7 nM T99041 CKY4R8 10112957 Ki = 281 nM T99041 CN5BD7 10114895 IC50 = 731 nM T99041 CIU12J 10116290 IC50 = 170 nM T99041 CM19YB 10125495 IC50 = 18000 nM T99041 CQT5Y2 10125644 IC50 = 1400 nM T99041 C10JOC 10125645 IC50 = 2500 nM T99041 CAOF95 10125896 IC50 = 200 nM T99041 C10BSW 10125952 IC50 = 1100 nM T99041 CD20SG 10125953 IC50 = 14000 nM T99041 CT6CG1 10126186 IC50 = 0.2 nM T99041 C0Q7BK 10127057 IC50 = 42 nM T99041 CNC5D4 10130367 Ki = 182 nM T99041 C9ERD7 10130575 IC50 = 22 nM T99041 CBL6T7 10132708 IC50 = 5 nM T99041 CLZF79 10133903 Ki = 12 nM T99041 C2RW5Z 10135822 Ki = 324 nM T99041 C4U3IC 10144962 IC50 = 139 nM T99041 C2H0UF 10149048 Ki = 0.03 nM T99041 C2YUP9 10149491 IC50 = 14000 nM T99041 CUE7K0 10156677 Ki = 112 nM T99041 C4CX1P 10157141 IC50 = 128 nM T99041 CUB1G7 10157334 Ki = 68 nM T99041 C6PZ1U 10160012 Ki = 316 nM T99041 C0L1KV 10162433 Ki = 428 nM T99041 C29RUO 10162817 Ki = 579 nM T99041 CQ3K8W 10164624 IC50 = 1900 nM T99041 C5X4NF 10171676 IC50 = 1000 nM T99041 C98FDL 10172375 IC50 = 0.9 nM T99041 C6SQ0P 10172376 IC50 = 90 nM T99041 CJ3MD2 10172601 IC50 = 100 nM T99041 C2SNQ8 10172681 IC50 = 240 nM T99041 C2KWM9 10172706 IC50 = 3 nM T99041 CXUC74 10173174 IC50 = 130 nM T99041 CKWE80 10176680 Ki = 2.2 nM T99041 C1UAG7 10176937 IC50 = 25 nM T99041 CEM94Y 10178009 IC50 = 539 nM T99041 C6S5OX 10179212 Ki = 29 nM T99041 CF7C3M 10180260 Ki = 45 nM T99041 C4FC2O 10183667 IC50 = 108 nM T99041 C7PWN9 10193213 IC50 = 31000 nM T99041 CWU9N2 10198228 Ki = 3 nM T99041 C05DXJ 10200731 Ki = 302 nM T99041 C6ISW4 10203198 Ki = 309 nM T99041 CD2U3A 10203599 Ki = 63 nM T99041 CQ8N1T 10209865 IC50 = 134 nM T99041 CFP27I 10214732 IC50 = 42000 nM T99041 C0CPY9 10215103 IC50 = 370 nM T99041 CL4T7Z 10215326 IC50 = 270 nM T99041 CLO81K 10215577 IC50 = 1750 nM T99041 C68WBI 10215628 IC50 = 47 nM T99041 CQ0V1C 10219838 IC50 = 39000 nM T99041 CZ9XN0 10220206 IC50 = 170 nM T99041 CBZ3P2 10221723 Ki = 56 nM T99041 CBC45I 10222923 Ki = 1278 nM T99041 CZ92XV 10225547 Ki = 76 nM T99041 CU9W8N 10233525 IC50 = 405 nM T99041 COD64C 10236556 IC50 = 47000 nM T99041 CYCJ68 10236557 IC50 = 1500 nM T99041 C9K3JS 10237877 IC50 = 180 nM T99041 C5P0AO 10238227 IC50 = 113 nM T99041 CTG4S9 10238900 IC50 = 1397 nM T99041 CCS75T 10242745 IC50 > 1000000 nM T99041 CW6PG0 10243173 Ki = 811 nM T99041 C07QCO 10243334 IC50 = 346 nM T99041 C6JS1Y 10245529 IC50 = 42 nM T99041 C0A9OY 10249393 IC50 = 30 nM T99041 CZ90LD 10250452 IC50 = 12 nM T99041 CU8C5K 10254918 IC50 = 5 nM T99041 C17HUN 10255762 IC50 = 8.4 nM T99041 C6ER9U 10269517 IC50 = 50 nM T99041 CQ07AR 10270647 Ki = 33 nM T99041 C9BPX2 10270831 IC50 = 280 nM T99041 CD0P5E 10271196 Ki = 530 nM T99041 CQ36IM 10272290 Ki = 24 nM T99041 C6M4SQ 10286219 IC50 = 1500 nM T99041 CAPB18 10286460 IC50 = 200 nM T99041 CZHS09 10286494 IC50 = 10000 nM T99041 CHWJ15 10286977 IC50 = 0.2 nM T99041 CT6FG8 10287141 IC50 = 340 nM T99041 C7AQS6 10287238 IC50 = 3 nM T99041 CHO8E7 10296151 Ki = 1 nM T99041 CC63ZN 10296260 IC50 = 864 nM T99041 CA7Q8J 10298482 Ki = 65 nM T99041 CY3LK8 10300368 Ki = 310 nM T99041 C9FZ2O 10304081 IC50 = 225 nM T99041 C8J3NA 10304145 IC50 = 44 nM T99041 C7US0V 10304855 IC50 = 114 nM T99041 CJDY62 10306170 IC50 = 14 nM T99041 C5AXF1 10308325 IC50 = 20000 nM T99041 CEGV15 10308355 IC50 = 40000 nM T99041 CNX7Q1 10308853 IC50 = 920 nM T99041 CTZN24 10309295 IC50 = 350 nM T99041 CQYE24 10309373 IC50 = 53 nM T99041 C3FB4T 10310021 IC50 = 91 nM T99041 CY6N9I 10318743 IC50 = 9.6 nM T99041 CF1S8U 10320144 IC50 = 4 nM T99041 C08UHI 10320529 IC50 = 117000 nM T99041 CC2TP8 10321088 IC50 = 5 nM T99041 CNV4R3 10324641 IC50 = 5.8 nM T99041 C0JD8Z 10333136 IC50 = 16 ug.mL-1 T99041 CIAV18 10333629 IC50 >> 1000000 nM T99041 CL72FC 10334538 IC50 > 1000000 nM T99041 C4UTO9 10336929 IC50 = 44 nM T99041 CM6Y1B 10339570 Ki = 5 nM T99041 CXP16T 10340933 IC50 = 15000 nM T99041 C1AEN6 10341846 IC50 > 125000 nM T99041 CEZ95L 10342016 IC50 = 58 nM T99041 CKZT43 10353699 IC50 = 518000 nM T99041 CU6LC2 10355512 IC50 = 104 nM T99041 CR0QC5 10367502 IC50 = 3 nM T99041 CP4M2R 10375745 IC50 = 80 nM T99041 CW70CV 10376453 IC50 >> 1000000 nM T99041 C7UO3L 10376704 Ki = 25 nM T99041 CK07VX 10376940 IC50 = 217000 nM T99041 CK8T4C 10381531 IC50 = 14.1 ug.mL-1 T99041 C79UAO 10381586 IC50 > 100 ug.mL-1 T99041 CQ7J2Z 10383508 IC50 = 15 nM T99041 C2GT0H 10384474 IC50 = 80 nM T99041 CY5M4R 10388027 IC50 = 26 nM T99041 CHZ85I 10393133 IC50 = 4800 nM T99041 CLI51Z 10398371 IC50 > 1000000 nM T99041 C29MEL 10399628 Ki = 22 nM T99041 C2EPA5 10401083 IC50 = 635 nM T99041 C6GWB8 10401570 IC50 > 100 ug.mL-1 T99041 C8NAX7 10403949 IC50 > 500000 nM T99041 CE0AS5 10405951 IC50 = 9 nM T99041 C7R6TZ 10406789 IC50 = 100 nM T99041 CVK1G5 10412922 IC50 = 13 nM T99041 CTK71I 10415171 IC50 = 400 nM T99041 C92DAJ 10415172 IC50 = 5600 nM T99041 C7F8SB 10420127 IC50 = 612 nM T99041 C7YIE3 10423532 Ki = 90 nM T99041 C1O2RY 10426457 IC50 = 11.5 nM T99041 C80ZBS 10429788 IC50 = 71 nM T99041 CUS9F6 10432611 IC50 = 13 nM T99041 C6GHF1 10433039 IC50 = 45 nM T99041 CWCA76 10439426 IC50 = 0.48 nM T99041 CAF71Y 10443207 IC50 = 247000 nM T99041 C4BKD9 10445283 Ki = 959 nM T99041 CO59EL 10450114 IC50 = 6.6 nM T99041 CCTY29 10451878 IC50 = 50 nM T99041 C4OC6P 10455620 IC50 = 175 nM T99041 C1WKE4 10455621 IC50 = 100 nM T99041 CHP37D 10456407 IC50 = 142000 nM T99041 C03IBO 10467163 Ki = 3800 nM T99041 CLV58Q 10468265 IC50 >> 1000000 nM T99041 CH1DG5 10478099 IC50 = 92 nM T99041 CL3H9I 10491923 IC50 > 100 ug.mL-1 T99041 CJ2RK6 10492044 IC50 > 100 ug.mL-1 T99041 CF46MR 10515590 IC50 = 70 nM T99041 C30TAX 10538170 IC50 = 95 nM T99041 CN4BI1 10564514 IC50 = 32 nM T99041 C8KLC3 10584166 IC50 = 11 nM T99041 CK3IW4 10584272 IC50 = 3500 nM T99041 C0KTQ5 10607253 IC50 = 50400 nM T99041 C38IDQ 10608000 IC50 = 250 nM T99041 C4PJ7H 10656779 Ki = 2150 nM T99041 C3YS4K 10659346 IC50 > 100 ug.mL-1 T99041 CN5KG9 10661540 IC50 = 12.8 ug.mL-1 T99041 CH6S5L 10704521 IC50 = 60 nM T99041 CXE71J 10750510 IC50 = 30000 nM T99041 CHA8X6 10751333 IC50 = 94000 nM T99041 CYLO09 10774283 IC50 = 52000 nM T99041 C1LSP2 10779050 IC50 > 100 ug.mL-1 T99041 CL26WQ 10780092 IC50 = 286000 nM T99041 C2KDY6 10798619 IC50 = 374000 nM T99041 C1WG0P 10798659 IC50 = 0.3 nM T99041 C1ZJ4I 10799226 IC50 = 107000 nM T99041 CJKX61 10821833 IC50 = 67000 nM T99041 C7BLJ1 10821834 IC50 > 1000000 nM T99041 CHC1X4 10824414 IC50 = 63 nM T99041 C3E8ID 10845163 IC50 = 15000 nM T99041 CK9SB4 10845727 IC50 = 93000 nM T99041 CCR8J7 10848386 IC50 = 17000 nM T99041 C04XQH 10850290 IC50 > 100 ug.mL-1 T99041 C1QL5M 10858831 IC50 > 1000000 nM T99041 C6QH7S 10860092 IC50 = 18600 nM T99041 C6WGA4 10861905 IC50 = 10 nM T99041 CJ39DG 10872395 IC50 > 500000 nM T99041 CS1LP6 10879478 IC50 = 24200 nM T99041 C3UGO0 10879937 IC50 = 53 nM T99041 C2QEW3 10883432 IC50 = 296 nM T99041 C4A5BM 10902702 IC50 = 598 nM T99041 C6ERS7 10904132 IC50 = 23 nM T99041 CVI2T1 10911918 IC50 = 103000 nM T99041 C42NLJ 10912330 IC50 = 7000 nM T99041 CV46YZ 10912691 IC50 = 33 nM T99041 CG9Q1Y 10923589 IC50 = 133 nM T99041 C9BL6G 10926029 IC50 = 70 nM T99041 CLA05J 10932707 Ki = 10 nM T99041 CPG58B 10943400 IC50 = 475 nM T99041 C6HNK4 10947008 IC50 = 7 nM T99041 CTWI82 10950467 IC50 = 149 nM T99041 CYP97B 10958030 IC50 = 17 nM T99041 CF60BW 10966961 IC50 = 26 nM T99041 CY9CW2 10969177 IC50 = 8 nM T99041 CW63DG 10980018 IC50 = 434000 nM T99041 C63VGB 10993665 IC50 = 64 nM T99041 CM5E1A 11000330 IC50 = 52600 nM T99041 CBFE09 11015514 IC50 = 183 nM T99041 CT9I8W 11020125 IC50 = 9610 nM T99041 CWR9G6 11023706 IC50 = 477000 nM T99041 CX1KF2 11024849 IC50 = 14 nM T99041 CA2OR9 11025044 IC50 = 228 nM T99041 CZ94WH 11025199 IC50 > 500000 nM T99041 C4MD5V 11037154 IC50 > 1000000 nM T99041 CH4TD3 11037548 IC50 = 326000 nM T99041 C0O8HF 11045633 IC50 = 29 nM T99041 CEPQ46 11053284 IC50 = 266 nM T99041 CTMK05 11056962 IC50 = 83 nM T99041 C42WCR 11065479 IC50 > 1000000 nM T99041 C9CYS1 11067211 IC50 = 931000 nM T99041 C9S8AG 11068388 IC50 = 16000 nM T99041 C0FWU4 11069462 IC50 = 22 nM T99041 CVJ81D 11075465 IC50 = 282 nM T99041 CNA61F 11076103 IC50 = 305 nM T99041 C60JXQ 11079321 IC50 > 1000000 nM T99041 C2N6MH 11084500 IC50 = 444 nM T99041 CX07LO 11085063 IC50 = 261 nM T99041 CSRO28 11089704 IC50 = 18 nM T99041 CS48RN 11098969 IC50 = 3000 nM T99041 COAR21 11101478 IC50 = 12000 nM T99041 CMO61N 11109983 IC50 = 338 nM T99041 C10CQP 11112644 IC50 = 62 nM T99041 CA4N0B 11117606 Ki = 11 nM T99041 C9GXD6 11117990 IC50 > 500000 nM T99041 C6QL3H 11122260 IC50 > 1000000 nM T99041 C1X8SI 11127914 IC50 = 398 nM T99041 CF41JX 11127915 IC50 = 105 nM T99041 CJB52P 11129932 IC50 = 3 nM T99041 CWDY68 11138020 IC50 = 192 nM T99041 C26ODF 11150893 IC50 > 500000 nM T99041 CXT8Y2 11151568 IC50 = 6 nM T99041 C4HBU9 11153488 IC50 = 30 nM T99041 CJ7E0N 11163434 IC50 = 0.13 nM T99041 CE94RO 11164254 IC50 = 9.3 nM T99041 C7HRW0 11164704 IC50 = 5 nM T99041 C82GSQ 11165177 IC50 = 77 nM T99041 CSB2T9 11166406 IC50 > 125000 nM T99041 CXR12G 11173505 Ki = 49 nM T99041 CX10UC 11173801 IC50 = 5.6 nM T99041 C5U1FY 11176598 IC50 = 830 nM T99041 CN3D5C 11180149 Ki = 0.59 nM T99041 CJS94B 11187292 IC50 = 5.6 nM T99041 C2ME1R 11187389 Ki = 8.9 nM T99041 CG49PR 11187940 Ki = 1.6 nM T99041 C9HKB7 11188314 IC50 = 23 nM T99041 C5E7VQ 11198004 IC50 = 20 nM T99041 CO9QM2 11198569 IC50 > 100000 nM T99041 CF1LD8 11199808 Ki = 0.4 nM T99041 C40SYQ 11200151 Ki = 8 nM T99041 C68XFD 11205761 IC50 > 1000000 nM T99041 C3BXS4 11206225 Ki = 14500 nM T99041 CMBT59 11207320 IC50 > 250000 nM T99041 CR60FN 11209195 IC50 = 17000 nM T99041 CW8FL2 11209569 IC50 = 301000 nM T99041 CJB87Z 11210511 IC50 = 9.7 nM T99041 C2PN1R 11211023 IC50 = 19 nM T99041 CH87RA 11211119 IC50 = 3.6 nM T99041 CHIZ26 11218348 IC50 = 6.3 nM T99041 C6VKT5 11219158 IC50 = 3700 nM T99041 CK5W4F 11220098 Ki = 143 nM T99041 CXAR72 11220471 IC50 = 250000 nM T99041 CSN6U7 11220682 IC50 = 18 nM T99041 CEUD41 11222126 IC50 = 2.6 nM T99041 CU3BG5 11222807 IC50 = 27 nM T99041 CJ2M8G 11222935 Ki = 1.4 nM T99041 C71YJO 11223701 Ki = 0.9 nM T99041 CK1UE7 11229192 IC50 = 188000 nM T99041 C35JSU 11229576 IC50 = 151000 nM T99041 C3X9SY 11229581 IC50 = 148000 nM T99041 CHX25W 11232123 IC50 = 345000 nM T99041 C0JD5Q 11232605 IC50 = 179000 nM T99041 CYL67P 11232890 Ki = 0.85 nM T99041 CR3PJ9 11233253 IC50 = 8 nM T99041 CVL7H4 11233695 IC50 = 30 nM T99041 C3UA7X 11234761 IC50 = 12 nM T99041 C32ZGY 11234800 IC50 = 3 nM T99041 CBES80 11235729 IC50 = 23 nM T99041 C5AB7G 11236208 IC50 = 1.49 nM T99041 C5CZH3 11242300 IC50 = 2130 nM T99041 CUS5G2 11243728 IC50 = 56000 nM T99041 CH82RJ 11244267 IC50 > 1000000 nM T99041 CDLT06 11245133 IC50 = 63 nM T99041 CQ6C5F 11246131 IC50 = 23 nM T99041 C4VQ0N 11246214 IC50 = 5 nM T99041 C67YUV 11253949 Ki = 3.9 nM T99041 CLJ7A1 11255193 IC50 = 417000 nM T99041 CR6N9B 11256457 IC50 = 430 nM T99041 C8M4XU 11256492 IC50 = 35 nM T99041 C2YS9G 11256520 IC50 = 5 nM T99041 C43HPD 11258527 IC50 = 990 nM T99041 C61KZW 11266019 IC50 = 496000 nM T99041 CN2O0L 11268786 IC50 = 4 nM T99041 CKL1A8 11268930 Ki = 0.93 nM T99041 CHO56W 11269281 IC50 = 570 nM T99041 CM0YI7 11269397 Ki = 0.96 nM T99041 C5IY0L 11269712 IC50 = 95000 nM T99041 CM1A5F 11270889 IC50 = 2.77 nM T99041 CR46GY 11277009 IC50 > 1000000 nM T99041 C17TLH 11277905 IC50 = 43 nM T99041 CXFV02 11278425 Ki = 3.5 nM T99041 CUB62P 11278798 IC50 = 4 nM T99041 CB5SD1 11280296 IC50 = 12 nM T99041 CUK58N 11281626 Ki = 0.4 nM T99041 CL5SH2 11281817 IC50 = 21 nM T99041 C0RWV3 11282205 IC50 = 7400 nM T99041 CWNT74 11283294 IC50 = 25 nM T99041 CUM48L 11288538 IC50 = 1.8 nM T99041 C0U2MV 11289193 IC50 = 205000 nM T99041 CO59DU 11289695 IC50 = 6.5 nM T99041 CTC0P9 11289792 IC50 = 148000 nM T99041 CM85DX 11291335 IC50 = 7800 nM T99041 C1YH5K 11291901 IC50 = 36 nM T99041 CCDX51 11292489 Ki = 3.8 nM T99041 CPD0L4 11292861 Ki = 0.35 nM T99041 CSH2N3 11294846 IC50 = 3 nM T99041 C51QAB 11300739 IC50 = 418000 nM T99041 CZV8P2 11300763 Ki = 10 nM T99041 CAL43D 11302841 IC50 = 13 nM T99041 C1TZY0 11302974 Ki = 42 nM T99041 CAW02M 11303089 IC50 = 14 nM T99041 CDZ79G 11304224 IC50 = 240 nM T99041 C2SOA8 11306467 IC50 = 71 nM T99041 CEJ32C 11306468 IC50 = 71 nM T99041 C06NLF 11309656 IC50 = 190000 nM T99041 C8I1QE 11310450 IC50 = 500000 nM T99041 C47GSV 11310499 IC50 = 23000 nM T99041 CP9LQ0 11312069 IC50 = 278000 nM T99041 CG8SA2 11312331 IC50 = 13 nM T99041 C4GUX3 11312733 IC50 > 500000 nM T99041 CMPH23 11313182 IC50 = 13 nM T99041 CEZ27P 11314348 Ki = 0.6 nM T99041 CM28RS 11314596 IC50 = 890 nM T99041 CL72NR 11314959 Ki = 0.45 nM T99041 CT6MF7 11316670 IC50 = 3 nM T99041 CTG12Q 11321743 IC50 = 23100 nM T99041 C9XYK1 11325183 IC50 = 6.2 nM T99041 CS8OH7 11326271 IC50 = 430 nM T99041 CK6G2V 11335782 Ki = 270 nM T99041 C43RXS 11337326 IC50 = 22 nM T99041 C38ADT 11346439 IC50 = 125000 nM T99041 C5SR4K 11346707 IC50 = 350 nM T99041 C9SJ0O 11347777 Ki = 607 nM T99041 CM4CT0 11348315 IC50 = 10 nM T99041 CM5E2A 11349317 IC50 = 57 nM T99041 C35GXU 11350142 Ki = 10 nM T99041 CNB7G8 11356095 IC50 = 39000 nM T99041 C24QLP 11356421 IC50 = 1000000 nM T99041 C1WOH9 11359214 IC50 > 500000 nM T99041 CK2T6J 11359671 IC50 = 17 nM T99041 CUH3S7 11360493 IC50 = 20 nM T99041 CQ9TJ5 11360810 IC50 = 3.7 nM T99041 CZ93VH 11361944 IC50 = 6 nM T99041 CKP0G9 11362130 IC50 = 34 nM T99041 CZ37IN 11372458 IC50 = 192000 nM T99041 CCNX41 11372959 IC50 = 540 nM T99041 CMZ1S9 11373129 IC50 = 6 nM T99041 CW3QZ7 11374531 IC50 = 19.4 nM T99041 C30JEU 11381416 IC50 = 69 nM T99041 C9FN7U 11381726 IC50 > 500000 nM T99041 CQ0MC7 11383372 IC50 = 200 nM T99041 CH74XT 11383468 IC50 > 500000 nM T99041 CE3O6K 11386357 IC50 = 14 nM T99041 CML13R 11389441 Ki = 7000 nM T99041 CH35IZ 11392716 IC50 = 14 nM T99041 CF01WK 11392988 Ki = 2.9 nM T99041 CL9HN3 11395030 Ki = 2 nM T99041 CD5A7Z 11395141 Ki = 10 nM T99041 CR9EB8 11396245 IC50 = 5 nM T99041 CEZS68 11403720 Ki = 28 nM T99041 CSR53F 11404106 IC50 = 186000 nM T99041 C0X6EK 11404881 Ki = 0.72 nM T99041 CI40EH 11405274 Ki = 57 nM T99041 C50PNA 11405365 Ki = 7.1 nM T99041 C3QZD5 11406220 Ki = 5.5 nM T99041 CTW02K 11406276 Ki = 0.67 nM T99041 CV1E7C 11406559 IC50 = 109 nM T99041 C3S8BD 11415118 IC50 = 5.6 nM T99041 C9AW7O 11416338 IC50 = 5 nM T99041 C0RIS4 11417008 IC50 = 15.1 nM T99041 CW8K3F 11417567 IC50 = 6.8 nM T99041 C2ZT0L 11418204 IC50 = 8 nM T99041 CRZ5F1 11418876 IC50 = 27 nM T99041 CFD62G 11419146 IC50 = 6 nM T99041 CPY7B2 11424308 Ki = 26 nM T99041 C3AZ7K 11426348 IC50 = 15 nM T99041 CB5C1T 11428334 Ki = 12 nM T99041 CY15PU 11429829 Ki = 0.83 nM T99041 CFTC85 11432169 IC50 = 29 nM T99041 C27ITV 11436930 IC50 = 250000 nM T99041 CLF89Y 11437087 IC50 > 1000000 nM T99041 CH39KX 11437726 IC50 = 188000 nM T99041 C82ENX 11439333 IC50 = 7 nM T99041 CRW3G4 11440163 IC50 = 10 nM T99041 CN9ZA8 11441300 IC50 = 68 nM T99041 CH09SE 11447824 IC50 > 1000000 nM T99041 CPNU92 11448828 IC50 = 4.9 nM T99041 CUG51Q 11449442 IC50 = 132000 nM T99041 C9RZC1 11450265 IC50 = 70000 nM T99041 CW27UK 11450266 IC50 = 500000 nM T99041 CZ68MT 11451290 IC50 = 8 nM T99041 CY0JG1 11451461 Ki = 1.6 nM T99041 C0DT1O 11451712 Ki = 7.4 nM T99041 CX5Y7J 11451739 Ki = 10 nM T99041 C6P2BR 11452943 Ki = 0.62 nM T99041 C6US2X 11461807 IC50 = 8 nM T99041 CV71FH 11464036 IC50 = 8 nM T99041 C1M9UX 11469862 Ki = 2.2 nM T99041 CWO06L 11471453 IC50 = 10 nM T99041 C7TOQ4 11472776 IC50 > 500000 nM T99041 CO7T4W 11473127 IC50 > 500000 nM T99041 C53RWU 11474019 IC50 = 266000 nM T99041 C6WT7P 11474308 Ki = 25 nM T99041 C5TQP7 11474372 Ki = 31 nM T99041 CE5A4M 11475797 IC50 = 34.3 nM T99041 C7JWD3 11476287 IC50 = 18 nM T99041 CS4H7X 11481506 Ki = 5.2 nM T99041 C6U9KB 11484559 IC50 = 4 nM T99041 C4G9AM 11484758 IC50 = 510 nM T99041 CPL64M 11486126 Ki = 21 nM T99041 CTD0S4 11486251 Ki = 0.98 nM T99041 CNMA97 11487118 IC50 = 128 nM T99041 CBV79P 11487883 Ki = 0.62 nM T99041 CEHI82 11493140 IC50 > 3000 nM T99041 C06RUA 11493219 IC50 = 64 nM T99041 C3MPY0 11493220 IC50 = 955 nM T99041 CDT16S 11493492 Ki = 28 nM T99041 CUTS18 11494449 IC50 = 2800 nM T99041 C50YHW 11494571 IC50 = 31300 nM T99041 C9PRY1 11494684 IC50 = 811 nM T99041 CJD30Y 11495704 IC50 = 2.3 nM T99041 CGA6Q4 11500119 IC50 = 4000 nM T99041 CAH5Z6 11500899 IC50 = 91 nM T99041 C2D9AT 11500939 Ki = 103 nM T99041 CKWZ03 11501743 IC50 = 80 nM T99041 CH7VS5 11505454 IC50 = 28 nM T99041 CBM01H 11507111 IC50 = 1600 nM T99041 CW38YC 11507527 IC50 = 89 nM T99041 C3XAT0 11507559 IC50 = 687 nM T99041 C62RBF 11507639 IC50 = 261 nM T99041 CF2S9Q 11507721 IC50 > 30000 nM T99041 C30JDP 11508177 IC50 = 1070 nM T99041 CLH62G 11508839 IC50 = 19 nM T99041 CM8QB3 11510166 Ki = 93 nM T99041 CQDM72 11514208 IC50 = 1000 nM T99041 C04OAE 11514331 IC50 = 1110 nM T99041 C7CLT9 11515196 IC50 = 118 nM T99041 CA3FS5 11515240 IC50 = 123 nM T99041 C15UQK 11515912 IC50 = 428 nM T99041 CO95FZ 11516000 IC50 = 1160 nM T99041 C0XVU3 11516085 IC50 = 7.6 nM T99041 C2S8BH 11516511 Ki = 14 nM T99041 CH5A7Q 11518007 IC50 = 2.5 nM T99041 C91OHR 11522044 IC50 > 3000 nM T99041 CJM1L9 11522376 IC50 = 62 nM T99041 C31ZBJ 11522467 IC50 = 689 nM T99041 C2TCM8 11523077 IC50 = 6.6 nM T99041 CY96CU 11523396 IC50 = 14800 nM T99041 CDCI64 11524392 IC50 = 14 nM T99041 C8KB4F 11524437 Ki = 612 nM T99041 CMYN65 11526865 IC50 = 150 nM T99041 C0O3XD 11527019 IC50 = 19 nM T99041 CWH3S0 11529375 IC50 = 52 nM T99041 CMN4Y5 11529427 IC50 = 1220 nM T99041 COL08I 11529539 IC50 = 97 nM T99041 CQ56DV 11529688 IC50 = 257 nM T99041 CXA53K 11529948 IC50 = 208 nM T99041 C10LHK 11531002 IC50 = 371 nM T99041 CV1N6Z 11531612 IC50 = 17 nM T99041 CZFI65 11531704 Ki = 30 nM T99041 C1B8JN 11532057 Ki > 10000 nM T99041 CZ35WN 11533932 IC50 = 13 nM T99041 C63DBH 11537823 Ki = 44 nM T99041 COXK41 11537890 Ki = 137 nM T99041 CKM89Z 11538673 IC50 = 22 nM T99041 CFXG35 11538686 IC50 = 13400 nM T99041 CMD6H8 11538715 IC50 = 5.8 nM T99041 CK36XC 11538961 Ki = 18 nM T99041 CG7I8Z 11538992 IC50 = 21 nM T99041 CPR71X 11540951 IC50 = 2.7 nM T99041 C98GDW 11541277 IC50 = 61 nM T99041 CBR9K8 11541314 IC50 = 7.5 nM T99041 CC5M2E 11544575 IC50 = 69 nM T99041 C1HV5Q 11544965 IC50 = 702 nM T99041 CVT52Y 11545508 IC50 = 30 nM T99041 C6KBN4 11546261 Ki = 2.2 nM T99041 CJIX61 11547698 IC50 = 9.9 nM T99041 C5AR6V 11550675 IC50 = 201 nM T99041 C9I5GV 11551088 IC50 = 26 nM T99041 C5NC3J 11551710 Ki = 21 nM T99041 CY3RK7 11551987 IC50 = 102 nM T99041 C6SA9R 11552616 IC50 = 25600 nM T99041 C2DJ6Y 11552953 Ki = 27 nM T99041 CA16WP 11554165 IC50 = 4.8 nM T99041 CCFP45 11558852 IC50 = 205 nM T99041 CV74GT 11559033 Ki = 143 nM T99041 C85EQW 11559371 IC50 = 50 nM T99041 CDK7I5 11559922 Ki = 0.4 nM T99041 CIZ52M 11561317 Ki = 11 nM T99041 CJF19H 11564906 IC50 = 663 nM T99041 CTE30Z 11565791 IC50 = 164 nM T99041 CL4D9A 11565911 IC50 = 66 nM T99041 CMN2K0 11566106 IC50 = 564 nM T99041 CI5W4Y 11566450 IC50 = 106 nM T99041 CLU15X 11566865 IC50 = 454 nM T99041 C4QG9W 11567318 Ki = 1310 nM T99041 CR37GC 11567606 Ki = 2.9 nM T99041 CAR0J5 11567905 IC50 = 24 nM T99041 CR4I1P 11568333 Ki = 4.4 nM T99041 CL41DG 11569450 Ki = 4.6 nM T99041 CY0A7J 11570138 IC50 = 4.3 nM T99041 CW4LO8 11572237 IC50 = 40000 nM T99041 CH76QT 11572962 IC50 = 8 nM T99041 C8G7UP 11573204 Ki = 49 nM T99041 CHL5Y0 11573374 IC50 = 875 nM T99041 C6F4OE 11573417 IC50 = 132 nM T99041 CAE39I 11573427 IC50 = 84 nM T99041 CCR9Q2 11574031 IC50 = 317 nM T99041 C25SEL 11574694 IC50 = 29 nM T99041 CE03TL 11574811 Ki = 28 nM T99041 CQU80H 11576569 IC50 = 55 nM T99041 C7P0NT 11576820 Ki = 54 nM T99041 CW94NS 11577331 IC50 = 8 nM T99041 CQ86GI 11577431 IC50 = 4.1 nM T99041 CJV39M 11579395 Ki = 377 nM T99041 CW31KG 11579932 IC50 = 61 nM T99041 C0T9NU 11580126 IC50 > 3000 nM T99041 C7BJK9 11580332 IC50 > 30000 nM T99041 C7EA6G 11580446 IC50 > 30000 nM T99041 CVG3B6 11580945 IC50 = 447 nM T99041 CCR0D7 11581247 IC50 = 83 nM T99041 CYT4Z1 11581458 IC50 = 49 nM T99041 CA4XU3 11581644 IC50 = 210 nM T99041 C9J1NO 11581694 IC50 = 24 nM T99041 CS6X0E 11581890 IC50 = 128 nM T99041 CAZL49 11584650 IC50 = 13 nM T99041 CUS2H6 11587911 IC50 > 3000 nM T99041 COH9V8 11589872 IC50 = 2.8 nM T99041 C5JYV7 11591936 IC50 = 8 nM T99041 CSCW37 11592154 IC50 = 2.6 nM T99041 CDE3P6 11594121 IC50 = 33 nM T99041 C3NT1E 11594414 IC50 = 160 nM T99041 CA51WQ 11595401 IC50 = 33 nM T99041 CI0E4X 11595565 Ki = 2.2 nM T99041 CO0QJ8 11596007 Ki = 1530 nM T99041 CE8M3K 11596123 Ki = 67 nM T99041 C9MXO0 11596219 IC50 = 116 nM T99041 CW48NY 11596451 Ki = 6.7 nM T99041 CMUV42 11596607 IC50 = 5.2 nM T99041 CSW3M9 11597271 IC50 = 6.9 nM T99041 C9SC1G 11602166 IC50 = 9400 nM T99041 CY4W0X 11602707 IC50 = 11 nM T99041 CHM2N0 11602713 Ki = 317 nM T99041 C9CM7N 11603627 IC50 = 18 nM T99041 CBE6K8 11603637 Ki = 22 nM T99041 CPXV24 11603996 IC50 = 17 nM T99041 C9N2EZ 11604004 Ki = 6.8 nM T99041 CGAF90 11604063 IC50 = 3059 nM T99041 CL4NM7 11604454 IC50 = 676 nM T99041 C0S2RQ 11605368 IC50 = 4.6 nM T99041 C15DLO 11608317 IC50 > 33000 nM T99041 C5V1XM 11608625 IC50 > 3000 nM T99041 C9JZM7 11608919 IC50 > 3000 nM T99041 C6I0XG 11609419 IC50 = 1500 nM T99041 COF62W 11611325 Ki = 9 nM T99041 CAOP57 11612570 IC50 = 715 nM T99041 CQL5S8 11613750 IC50 = 6.2 nM T99041 CZ91WO 11616288 IC50 = 630 nM T99041 C27JCR 11616775 IC50 = 13600 nM T99041 C6MO9K 11616857 IC50 = 651 nM T99041 CD3YU1 11616861 IC50 = 74 nM T99041 CEX4O6 11617338 IC50 = 54 nM T99041 C7KS2Q 11617492 IC50 = 600 nM T99041 C40ZJT 11619382 IC50 = 73 nM T99041 C2APG7 11623550 IC50 = 72 nM T99041 CR8XO2 11623606 IC50 = 59 nM T99041 C7QC6U 11623777 Ki = 1280 nM T99041 C17XSP 11623929 Ki = 8.3 nM T99041 CPSN73 11624012 Ki = 20 nM T99041 CH2JP9 11624034 IC50 > 30000 nM T99041 CDZ72J 11624893 IC50 = 1108 nM T99041 CRY2D5 11625412 Ki = 50 nM T99041 C7YKC0 11628195 IC50 = 22 nM T99041 C5AKH1 11630368 IC50 = 2000 nM T99041 CYR61O 11630666 IC50 = 320 nM T99041 CV17GF 11631125 IC50 = 66 nM T99041 CA1J8U 11631434 IC50 = 3300 nM T99041 CH3WM8 11632024 IC50 = 8400 nM T99041 CSO1D6 11632159 Ki = 43 nM T99041 CZT57X 11632256 IC50 = 52 nM T99041 C8Y3FM 11632315 IC50 = 29 nM T99041 CM1DR9 11632375 Ki = 22 nM T99041 C09KAV 11632502 IC50 = 17 nM T99041 C7SP9Y 11634778 Ki > 3000 nM T99041 CR6NM8 11638575 Ki = 33 nM T99041 CM6QE9 11638687 IC50 > 3000 nM T99041 CHLA97 11638762 Ki = 241 nM T99041 CRA0H5 11639131 Ki = 550 nM T99041 C0M1HR 11640120 IC50 = 4.8 nM T99041 C5P3NB 11644467 IC50 = 56 nM T99041 C3RZO9 11645337 IC50 = 452 nM T99041 CQO8U6 11648011 Ki > 10000 nM T99041 CXG1B4 11649741 IC50 = 6.3 nM T99041 CO2YH1 11652954 Ki = 764 nM T99041 C1Y2DC 11652956 Ki = 867 nM T99041 CZBD50 11653749 Ki = 96 nM T99041 C94OMG 11654093 Ki = 18 nM T99041 C8AU5P 11654528 Ki = 38 nM T99041 CUX2M0 11654810 Ki = 7.2 nM T99041 C52ION 11655271 Ki = 19 nM T99041 CT4W8K 11659101 IC50 = 790 nM T99041 C7M6ZY 11659120 IC50 = 45200 nM T99041 CR8Z6I 11659133 IC50 > 30000 nM T99041 CZFV81 11661472 IC50 = 260 nM T99041 CI8EF3 11666622 IC50 > 3000 nM T99041 CN3WA7 11668525 IC50 > 3000 nM T99041 CE91WR 11669357 IC50 = 20 nM T99041 C43OVS 11673852 IC50 = 96 nM T99041 CCBS09 11674180 Ki = 64 nM T99041 CH1KG5 11674534 IC50 = 57 nM T99041 CTNO72 11674721 IC50 = 4.6 nM T99041 C2G6RP 11675637 Ki = 75 nM T99041 CI1ED9 11676224 IC50 = 150 nM T99041 C3Y7EL 11678025 IC50 = 5.2 nM T99041 C1A7NS 11680394 IC50 = 98 nM T99041 C5BD4Q 11680960 Ki = 12 nM T99041 CV0XW8 11680991 IC50 = 298 nM T99041 CFX6Z9 11681207 IC50 = 32 nM T99041 CNF1M4 11681778 IC50 = 50 nM T99041 C2K9XG 11688776 IC50 = 10 nM T99041 C0IWC9 11689866 IC50 = 651 nM T99041 CA69TN 11690566 IC50 = 77 nM T99041 C8UYQ5 11690713 IC50 = 2500 nM T99041 CC9O1L 11692537 Ki = 0.27 nM T99041 CEAN27 11694995 Ki = 1610 nM T99041 CBW6A1 11695523 IC50 = 6300 nM T99041 C79ECL 11695535 IC50 = 3236 nM T99041 C45QIU 11695818 IC50 = 2800 nM T99041 C7DCV9 11696495 Ki = 438 nM T99041 C6JPE0 11696912 Ki = 495 nM T99041 CRU2Q1 11697286 Ki = 5.6 nM T99041 C2WK1Z 11697387 Ki = 20 nM T99041 C1KCR6 11702577 IC50 = 15000 nM T99041 C2F6BA 11702880 Ki = 15 nM T99041 C8SI4E 11702902 IC50 = 119 nM T99041 C0Q3IL 11703158 IC50 = 784 nM T99041 C8IQA2 11703413 IC50 = 90 nM T99041 CUJ07L 11703663 Ki = 720 nM T99041 CJP1U8 11703749 IC50 = 1.5 nM T99041 C2X5GC 11704411 Ki = 9 nM T99041 C6YHK3 11704412 Ki = 24 nM T99041 CFO63Q 11704578 IC50 = 527 nM T99041 C1MGA4 11705197 Ki = 2.7 nM T99041 C8LA3E 11705712 Ki = 76 nM T99041 CU8LZ4 11705859 IC50 = 1418 nM T99041 CUC0Z3 11708771 IC50 = 400 nM T99041 CZF5D9 11708829 IC50 = 63 nM T99041 CNG85M 11710587 Ki = 8.9 nM T99041 CK4I6J 11710700 Ki = 6 nM T99041 C0CG5R 11710963 IC50 = 42 nM T99041 C04OMI 11711314 Ki = 113 nM T99041 C8VC2D 11711413 Ki = 33 nM T99041 C8KD6N 11711414 Ki = 163 nM T99041 C0U7QC 11715518 IC50 = 105 nM T99041 C34BEP 11716483 Ki = 12 nM T99041 CMI90R 11716843 Ki = 3.4 nM T99041 CCR80L 11717090 IC50 = 116 nM T99041 CZS71R 11717268 IC50 = 369 nM T99041 C1XD5I 11718004 Ki = 113 nM T99041 C1M7PL 11718857 Ki = 30 nM T99041 CY1S3Q 11719625 IC50 = 2.8 nM T99041 C0UJ7G 11719823 IC50 = 910 nM T99041 CIEJ54 11720809 IC50 = 5.3 nM T99041 CHA7Z9 11722557 IC50 = 119 nM T99041 CIOY84 11723708 IC50 = 21.3 ug.mL-1 T99041 C6VG7O 11727562 IC50 = 989 nM T99041 CJ6XR8 11730284 IC50 > 125000 nM T99041 CX9U4G 11731880 IC50 = 503000 nM T99041 C96TGJ 11746838 IC50 = 988 nM T99041 CA2H1U 11747757 IC50 = 163 nM T99041 C3ZPG6 11772582 IC50 = 68 nM T99041 CX84PY 11772583 IC50 = 590 nM T99041 C1P9ZM 11776124 IC50 > 1000000 nM T99041 C6JY7V 11776638 Ki = 8 nM T99041 CS0WM6 11778955 IC50 = 320 nM T99041 C3MX2I 11781105 IC50 = 24 nM T99041 CO73AL 11784400 IC50 = 15000 nM T99041 CKTJ04 11791651 IC50 = 291 nM T99041 C67TXV 11791652 IC50 = 109000 nM T99041 C1P2AI 11809137 IC50 = 102 nM T99041 C6ET2R 11817181 IC50 = 43500 nM T99041 CK24XY 11819467 IC50 > 1000000 nM T99041 C19HAP 11825584 IC50 = 89000 nM T99041 CN79VL 11840913 Ki = 6.7 nM T99041 CSOC43 11840914 Ki = 0.82 nM T99041 CE6V2H 11840916 Ki = 3.8 nM T99041 C42BOS 11854299 IC50 = 56.9 nM T99041 C2FN7G 11854301 IC50 = 53.4 nM T99041 CQ0O5A 11952574 IC50 = 120 nM T99041 CQIB43 11957945 IC50 = 82 nM T99041 CTQI92 11974546 Ki = 45 nM T99041 C5BZW6 11998979 Ki = 140 nM T99041 CXHC16 11999086 Ki = 240 nM T99041 CU3HD8 11999088 Ki = 190 nM T99041 CLI17Z 11999090 Ki = 220 nM T99041 C8U5NY 11999093 Ki = 15 nM T99041 CBZ03A 11999206 Ki = 76 nM T99041 C2TAJ9 11999207 Ki = 200 nM T99041 C3E4ZB 11999208 Ki = 34 nM T99041 C6DK9R 11999211 Ki = 35 nM T99041 CQSP03 12043866 IC50 = 207000 nM T99041 C35DEQ 12043867 IC50 = 3400 nM T99041 C1P3MJ 12043868 IC50 = 18000 nM T99041 C7NRQ3 12043869 IC50 = 731000 nM T99041 CAI8E7 12043870 IC50 = 51400 nM T99041 C21PAF 12069363 IC50 = 0.6 nM T99041 CQY50P 12742483 IC50 = 250000 nM T99041 C9RA7N 13478499 Ki = 160000 nM T99041 CYV1F7 13784835 IC50 > 100 ug.mL-1 T99041 C1GF7B 13939278 IC50 = 750 nM T99041 C94FPE 14434173 IC50 > 100 ug.mL-1 T99041 CR8H4L 14978092 IC50 = 200 nM T99041 CJAE28 15036410 IC50 = 118000 nM T99041 C6BHJ9 15101668 IC50 > 1000000 nM T99041 C29IHT 15337406 IC50 = 16000 nM T99041 CNM5V2 15940321 IC50 = 32360 nM T99041 C2ZMH8 15948988 IC50 = 25.4 nM T99041 C13JIX 15949418 IC50 = 0.67 nM T99041 C49NUJ 15949507 IC50 = 5.3 nM T99041 CPD3V1 15949508 IC50 = 0.5 nM T99041 CU4P5X 15950383 Ki = 3 nM T99041 C16XRI 15950384 Ki = 51.5 nM T99041 CUMR27 15950385 Ki = 11 nM T99041 C69RAY 15950386 Ki = 9 nM T99041 CM63YP 15950387 Ki = 29 nM T99041 CH8F7W 15950388 Ki = 4 nM T99041 C0L4SH 15950456 Ki = 14 nM T99041 C8G7OJ 15950457 Ki = 12 nM T99041 C8FU1V 15950462 Ki = 29 nM T99041 C9KJ6D 15950538 Ki = 2.7 nM T99041 C3C6PM 15950539 Ki = 9 nM T99041 C4S7AB 15950540 Ki = 4 nM T99041 C2HGJ0 15950541 Ki = 16 nM T99041 C3U1VO 15950542 Ki = 9 nM T99041 CKX8M6 15950615 Ki = 4 nM T99041 CC0M2X 15951427 Ki = 8 nM T99041 CF3PX0 15951428 Ki = 30 nM T99041 CWTX01 15951429 Ki = 12 nM T99041 C3LQD9 15951431 Ki = 18 nM T99041 C8M0FT 15951543 IC50 = 27 nM T99041 CI3DB4 15951636 IC50 > 20000 nM T99041 C3SM4T 15951642 IC50 > 100000 nM T99041 C8QRV9 15951839 Ki = 38400 nM T99041 CMNT83 15951928 Ki = 608000 nM T99041 CL1E6O 15953860 IC50 = 17 nM T99041 CG2E3Z 15991577 IC50 = 84 nM T99041 CLG2Q1 16035093 IC50 = 24 nM T99041 CMUG74 16035094 IC50 = 25 nM T99041 CYPG43 16040279 Ki = 3.2 nM T99041 C13-MAR 16040457 IC50 > 100000 nM T99041 C0YQ9A 16046127 IC50 = 325000 nM T99041 C75ZNE 16058650 Ki = 4 nM T99041 C28IRJ 16064807 IC50 = 17 nM T99041 C4LJH3 16064808 IC50 = 24 nM T99041 CVIC15 16064809 IC50 = 11 nM T99041 CS7DQ3 16090844 Ki = 3 nM T99041 C8CVG9 16090856 Ki = 1.3 nM T99041 CB6WK0 16121107 Ki = 170000 nM T99041 CZQ8O9 16121199 Ki = 100000 nM T99041 C5Q9BH 16122596 IC50 = 16 nM T99041 CU3GB5 16126742 IC50 = 4.8 nM T99041 CUQT90 16202787 Ki = 12 nM T99041 CHUX72 16202788 Ki = 3.8 nM T99041 C8D2RM 16203032 Ki = 1400 nM T99041 CW0JF5 16203033 Ki = 17 nM T99041 C5F6DE 16203034 Ki = 590 nM T99041 C0LJA8 16203036 Ki = 105 nM T99041 CC20IT 16203037 Ki = 4 nM T99041 CW6AC3 16203151 Ki = 6 nM T99041 C5BE1I 16204461 Ki = 1600 nM T99041 CWY50B 16204462 Ki = 930 nM T99041 CAQ7S4 16204463 Ki = 440 nM T99041 CCW34I 16204464 Ki = 270 nM T99041 CCWF31 16204465 Ki = 83 nM T99041 C73HLC 16204466 Ki = 24 nM T99041 CA1PV5 16216352 IC50 > 33000 nM T99041 CD9MQ6 16223559 IC50 = 245 nM T99041 CQ7G8T 16223560 IC50 = 1.7 nM T99041 CN24YP 16223762 IC50 = 984 nM T99041 CF37TH 16226604 IC50 = 84 nM T99041 C6ANU2 16226605 IC50 = 109 nM T99041 CFW43X 16658022 IC50 = 5 nM T99041 C6H5VO 16658023 IC50 = 5 nM T99041 CC9W4S 16658024 IC50 = 15 nM T99041 CR51WX 16658101 IC50 = 13 nM T99041 CMLR19 16658102 IC50 = 5 nM T99041 CXN32U 16658103 IC50 = 8 nM T99041 C2XP7B 16658104 IC50 = 4 nM T99041 CD6L7Z 16658105 IC50 = 19 nM T99041 C63NWG 16658243 IC50 < 10 nM T99041 C82ZAL 16658881 IC50 = 460 nM T99041 C24NZK 16658917 Ki = 2.3 nM T99041 C28GEM 16662696 IC50 = 1.1 nM T99041 C53XZP 16721117 Ki = 2 nM T99041 CW62MC 16725327 IC50 = 1.3 nM T99041 C0EV4T 16725905 IC50 = 5 nM T99041 C56LTN 16739329 IC50 = 0.92 nM T99041 CT01PQ 16739331 IC50 = 70 nM T99041 C19UBP 16747699 IC50 = 13 nM T99041 C9JK5Q 16750059 Ki = 5.3 nM T99041 C61RFP 16755651 Ki = 13 nM T99041 C4RK2Q 17591662 IC50 = 94.82 nM T99041 CU05RG 17748274 IC50 = 16 nM T99041 C15TBF 17751406 IC50 = 15000 nM T99041 C5W3VY 17753031 IC50 = 76 nM T99041 CX5F2U 17763521 IC50 > 500000 nM T99041 CQG89Z 17853548 IC50 = 41400 nM T99041 C6L7MA 18391459 IC50 = 2.9 nM T99041 CV4Z6Q 18398587 IC50 = 134900 nM T99041 CP3S0V 18398588 IC50 = 247000 nM T99041 C7GDU9 20038035 IC50 > 100 ug.mL-1 T99041 CC8RN3 20198196 IC50 = 18100 nM T99041 CT42AI 20706081 IC50 = 330 nM T99041 CBZ1E6 21045424 IC50 = 765 nM T99041 C6ZMS8 21054400 Ki = 5 nM T99041 CWB93R 21054485 IC50 = 21 nM T99041 CBY6M2 21919450 IC50 = 142 nM T99041 CH7YL4 21919455 IC50 = 10000 nM T99041 C1PF7M 21919463 IC50 = 2200 nM T99041 C39STQ 21919469 IC50 = 1150 nM T99041 C2OXL1 21919478 IC50 = 13 nM T99041 CY8OJ7 21947630 IC50 = 26 nM T99041 CQ9LB5 21947637 IC50 = 89 nM T99041 CCFX26 21947643 IC50 = 7 nM T99041 C3SXF7 21947646 IC50 = 4 nM T99041 CPES59 21949259 IC50 = 190000 nM T99041 C2W4KV 21949272 IC50 = 67000 nM T99041 CZ9K4Q 22029435 IC50 = 580 nM T99041 C0X4SO 22029457 IC50 = 340 nM T99041 CLK4G6 22029894 IC50 = 1230 nM T99041 C6BME5 22175258 IC50 = 1100 nM T99041 CRA87P 22175262 IC50 = 360 nM T99041 C7E0NG 22175290 IC50 = 2400 nM T99041 C2SD9C 22175298 IC50 = 2400 nM T99041 CQ3EB8 22175361 IC50 = 47 nM T99041 C56RIP 22175474 IC50 = 1900 nM T99041 C28HMT 22175479 IC50 = 1100 nM T99041 CK4NR7 22175497 IC50 = 1200 nM T99041 C2ME4A 22175534 IC50 = 870 nM T99041 C2RM7H 22175568 IC50 = 980 nM T99041 C7X5DS 22175618 IC50 = 3800 nM T99041 CE3LM6 22175639 IC50 = 250 nM T99041 CLUH89 22175659 IC50 = 4000 nM T99041 C4AUK1 22175709 IC50 = 8300 nM T99041 C6KGB8 22175713 IC50 = 220 nM T99041 CBYP16 22175758 IC50 = 250 nM T99041 CB38EC 22176094 IC50 = 1500 nM T99041 CR23XQ 22176165 IC50 = 2400 nM T99041 C8QF7T 22176298 IC50 = 1900 nM T99041 CUND82 22176405 IC50 = 1600 nM T99041 CL68SA 22220623 IC50 = 80000 nM T99041 C2XAR9 22401333 IC50 > 100000 nM T99041 CED47V 22690988 IC50 = 24000 nM T99041 C9VGC8 22691359 IC50 > 100000 nM T99041 C43XCK 22691633 Ki = 5300 nM T99041 C1M2ZS 22691666 IC50 > 100000 nM T99041 CM4SH2 23595882 IC50 = 167000 nM T99041 CP1J3T 23596395 Ki = 14 nM T99041 C8JSI4 23628284 IC50 = 50 nM T99041 CC29GD 23633277 IC50 = 0.5 nM T99041 C1RV7P 23633348 IC50 = 17 nM T99041 CU1LK3 23633350 IC50 = 1.5 nM T99041 CKN67W 23633553 IC50 = 6 nM T99041 CG37EL 23633557 IC50 = 7 nM T99041 C5U3NL 23633697 IC50 = 9 nM T99041 CVC80Z 23633837 IC50 = 10 nM T99041 C8P9GL 23633839 IC50 = 400 nM T99041 C5UVZ9 23634061 IC50 = 60 nM T99041 C5ZF2X 23634210 IC50 = 25 nM T99041 C4KW2T 23634279 IC50 = 4 nM T99041 CVF78O 23634281 IC50 = 4 nM T99041 CA95UP 23634434 IC50 = 8.4 nM T99041 C7FSW5 23634528 IC50 > 36900 nM T99041 CAQ81M 23644660 IC50 = 455 nM T99041 CDPU25 23644665 IC50 = 7360 nM T99041 CCSU21 23645371 IC50 = 27 nM T99041 C5M6UX 23645373 Ki = 470 nM T99041 CFS6P4 23645374 Ki = 20 nM T99041 CAVN39 23645375 Ki = 26 nM T99041 CN0FR1 23645376 Ki = 3.1 nM T99041 CVQ39W 23645377 Ki = 5.3 nM T99041 CQPA42 23645378 Ki = 36 nM T99041 CQ5R2G 23645379 Ki = 360 nM T99041 C32KIA 23645380 Ki = 1160 nM T99041 C6TCN1 23645381 Ki > 12800 nM T99041 CL08ZV 23645382 Ki > 12800 nM T99041 C8P3OQ 23645383 Ki > 12800 nM T99041 C72KLP 23645384 Ki = 980 nM T99041 CNVP26 23645385 Ki = 360 nM T99041 C3OHM9 23645386 Ki = 310 nM T99041 C8TP3W 23645387 Ki = 166 nM T99041 CZXL64 23645388 Ki = 160 nM T99041 C7MAX0 23645389 Ki = 170 nM T99041 C7W6PC 23645390 Ki = 96 nM T99041 CX0VJ4 23645391 Ki = 8900 nM T99041 C4EM3K 23645392 Ki > 12800 nM T99041 CU76EP 23645393 Ki > 12800 nM T99041 CFV07G 23645410 IC50 = 231 nM T99041 CIMG82 23645411 IC50 = 68 nM T99041 C47OZL 23645510 IC50 = 520 nM T99041 C2Q5IK 23645581 IC50 = 48 nM T99041 C3VA0M 23645582 IC50 = 968 nM T99041 C1JAG6 23645622 IC50 = 110 nM T99041 CDL4G9 23645678 Ki = 2.1 nM T99041 CL1DC7 23645680 Ki = 1.8 nM T99041 C23BMA 23645681 IC50 = 170000 nM T99041 C4B9FM 23645685 Ki = 1 nM T99041 CP9GS5 23645686 IC50 = 19700 nM T99041 C6R2LP 23645687 IC50 = 1820 nM T99041 CN7FK3 23645688 IC50 = 12400 nM T99041 CSHX17 23645689 IC50 = 4790 nM T99041 CL8QV6 23645690 IC50 = 4820 nM T99041 C0AU9X 23645691 IC50 = 990 nM T99041 CRM3Y4 23645692 IC50 = 15600 nM T99041 CDM8A2 23645693 IC50 = 3820 nM T99041 CIR1F6 23645694 IC50 = 1790 nM T99041 CK5G6I 23645695 IC50 = 1610 nM T99041 CHS76O 23645696 IC50 = 330 nM T99041 CVP59D 23645697 IC50 = 190 nM T99041 CH13BW 23645698 IC50 = 122 nM T99041 CL0K1T 23645699 IC50 = 520 nM T99041 CB3Z7O 23645700 IC50 = 4590 nM T99041 CNO6Q1 23645702 IC50 = 160 nM T99041 CGMC54 23645703 IC50 = 830 nM T99041 C0V4WR 23645705 IC50 = 43 nM T99041 CY9XW5 23645721 IC50 = 40 nM T99041 C5MO2Q 23645882 Ki = 260 nM T99041 C1UR3L 23645883 Ki = 507 nM T99041 C5EQ1C 23645884 Ki > 10000 nM T99041 CO90SF 23645885 Ki = 212 nM T99041 C85TUY 23645886 Ki = 1311 nM T99041 CBNC76 23645887 Ki = 140 nM T99041 CE1H2R 23645888 Ki = 513 nM T99041 CR7C8Q 23645889 Ki > 10000 nM T99041 CSW5F3 23645890 Ki = 4422 nM T99041 C7E8AI 23645891 Ki > 10000 nM T99041 C8YGE5 23645892 Ki = 399 nM T99041 C31TSP 23645893 Ki > 10000 nM T99041 C87LMT 23645894 Ki > 10000 nM T99041 CX79LQ 23645895 Ki = 74 nM T99041 CON27H 23645896 Ki = 27 nM T99041 CAYT68 23645897 Ki = 673 nM T99041 C5SH6W 23645898 Ki = 37 nM T99041 CDFZ57 23645899 Ki = 188 nM T99041 C5XB6V 23645900 Ki > 10000 nM T99041 CS6WQ4 23645901 Ki = 18 nM T99041 C9AZD2 23645902 Ki = 3 nM T99041 C2O6ML 23645903 Ki = 23 nM T99041 CKM6Y8 23645917 IC50 = 250 nM T99041 C9Y2ZL 23645918 IC50 = 110 nM T99041 C4V6BX 23645919 IC50 = 130 nM T99041 C78PNU 23645920 IC50 = 150 nM T99041 C5YT6S 23645921 IC50 = 180 nM T99041 CELQ89 23645922 IC50 = 150 nM T99041 CGV92H 23645923 IC50 = 350 nM T99041 CJ60EH 23645924 IC50 = 160 nM T99041 CZG70A 23645925 IC50 = 160 nM T99041 CD6V7X 23645926 IC50 = 220 nM T99041 C1TD4J 23645927 IC50 = 300 nM T99041 C71PQU 23645928 IC50 = 270 nM T99041 C8EOB9 23645929 IC50 = 780 nM T99041 C0M1TH 23645930 IC50 = 150 nM T99041 CFHB36 23645931 IC50 = 130 nM T99041 CTG27F 23645932 IC50 = 39 nM T99041 CS2FT5 23645933 IC50 = 72 nM T99041 C98QGK 23645934 IC50 = 160 nM T99041 CS76DY 23645935 IC50 = 130 nM T99041 C91MYK 23645936 IC50 = 85 nM T99041 C3AQC0 23645937 IC50 = 590 nM T99041 C61GTC 23645938 IC50 = 480 nM T99041 C8XF6R 23645939 IC50 = 310 nM T99041 C7IX5B 23645940 IC50 = 360 nM T99041 CP6M3W 23645941 IC50 = 260 nM T99041 CQ75XK 23645942 IC50 = 380 nM T99041 C8T7GY 23645943 IC50 = 130 nM T99041 C25ZXC 23645944 IC50 = 290 nM T99041 C4A3NI 23645945 IC50 = 180 nM T99041 C9Y1BP 23646016 IC50 = 73 nM T99041 CL8DY2 23646017 IC50 = 73 nM T99041 CT6Q1R 23646018 IC50 = 72 nM T99041 C8VS1X 23646019 IC50 = 144 nM T99041 CL4BX5 23646020 IC50 = 4130 nM T99041 CZ24WC 23646021 IC50 = 1957 nM T99041 C98VYW 23646022 IC50 = 2587 nM T99041 CCL17M 23646023 IC50 = 228 nM T99041 CT16HE 23646024 IC50 = 129 nM T99041 CAL8T5 23646025 IC50 = 63 nM T99041 CVSH12 23646026 IC50 = 274 nM T99041 C15HJB 23646027 IC50 > 100000 nM T99041 CBUM54 23646029 IC50 > 100000 nM T99041 C32ZNH 23646030 IC50 = 31000 nM T99041 CE8L2I 23646031 Ki = 64 nM T99041 C8SIU2 23646032 IC50 > 100000 nM T99041 C7L6JR 23646033 IC50 > 100000 nM T99041 CJ9ZL3 23646080 IC50 > 1000000 nM T99041 C0S2UB 23646081 IC50 > 1000000 nM T99041 CQ3KF6 23646082 IC50 > 1000000 nM T99041 CZ9P0Q 23646083 IC50 > 1000000 nM T99041 CFPN10 23646084 IC50 > 1000000 nM T99041 C0NV1B 23646085 IC50 > 1000000 nM T99041 CSW9T1 23646086 IC50 > 250000 nM T99041 CH72RP 23646087 IC50 > 1000000 nM T99041 CH5Y2F 23646088 IC50 > 500000 nM T99041 CJ47OR 23646089 IC50 > 250000 nM T99041 CRT2B0 23646090 IC50 > 250000 nM T99041 C7JXN0 23646091 IC50 > 1000000 nM T99041 C4K1NE 23646092 IC50 > 250000 nM T99041 CJV2K1 23646093 IC50 > 250000 nM T99041 C51BSR 23646094 IC50 > 250000 nM T99041 C2WDG4 23646095 IC50 > 125000 nM T99041 CB2ZT7 23646096 IC50 > 1000000 nM T99041 COF57U 23646097 IC50 > 1000000 nM T99041 CU26YP 23646098 IC50 > 250000 nM T99041 CM37ZS 23646100 IC50 > 1000000 nM T99041 C4SV2J 23646101 IC50 > 1000000 nM T99041 CX68KV 23646102 IC50 > 1000000 nM T99041 CZ28UC 23646142 Ki = 62 nM T99041 CLA15H 23646143 Ki = 4 nM T99041 C0EK5I 23646441 IC50 = 7.2 nM T99041 CF1TP9 23646442 IC50 = 160 nM T99041 CZA78Q 23646443 IC50 = 89 nM T99041 C5VP2I 23646444 IC50 = 14 nM T99041 C9PW1E 23646445 IC50 = 150 nM T99041 CAI0B5 23646446 IC50 = 2300 nM T99041 C4XM2W 23646447 IC50 = 67000 nM T99041 CUZ0D8 23646448 IC50 = 142 nM T99041 C7PE0S 23646449 IC50 = 16 nM T99041 COT87G 23646450 IC50 = 0.91 nM T99041 CF2J9Q 23646451 IC50 = 0.49 nM T99041 CVHU93 23646508 Ki = 9 nM T99041 CJLP47 23646509 Ki = 10 nM T99041 C7P5TW 23646510 Ki = 22 nM T99041 C61FRE 23646511 Ki = 1200 nM T99041 C4EG5D 23646512 Ki = 11 nM T99041 CN47RA 23646513 Ki = 29 nM T99041 CDM3J0 23646514 Ki = 25 nM T99041 CW0J6X 23646515 Ki = 57 nM T99041 CS6L8X 23646516 Ki = 300 nM T99041 COPD36 23646517 Ki = 260 nM T99041 CWT7X1 23646518 Ki = 450 nM T99041 C5GQ7J 23646519 Ki = 11 nM T99041 C0E8SM 23647079 IC50 = 280 nM T99041 CA6X5F 23647080 IC50 = 39 nM T99041 CP2W3B 23647081 IC50 = 3800 nM T99041 CS8O6P 23647082 IC50 = 820 nM T99041 CA53BK 23647084 IC50 = 110 nM T99041 CK15XF 23647085 IC50 = 340 nM T99041 CFOA63 23647106 IC50 = 13 nM T99041 CRF32I 23647107 IC50 = 5 nM T99041 CFTW63 23647114 IC50 = 20.7 nM T99041 C0BQ2D 23647115 IC50 = 11.6 nM T99041 CLO1Y2 23647116 IC50 = 69.9 nM T99041 CSJ78F 23647117 IC50 = 9 nM T99041 CDE9L7 23647118 IC50 = 11.5 nM T99041 CZF25M 23647119 IC50 = 15.1 nM T99041 CW5U3C 23647120 IC50 = 10.5 nM T99041 CWO62C 23647121 IC50 = 19.2 nM T99041 C0X1CK 23647122 IC50 = 8 nM T99041 C7JOV9 23647123 IC50 = 33 nM T99041 C0UT7J 23647124 IC50 = 397 nM T99041 C8P2VJ 23647125 IC50 = 37.3 nM T99041 CQ85KB 23647126 IC50 = 60.3 nM T99041 CRFL12 23647127 IC50 = 24.6 nM T99041 CP3CF0 23647128 IC50 = 143 nM T99041 CJA3M7 23647129 IC50 = 142 nM T99041 C7L3RX 23647130 IC50 = 11 nM T99041 C8UWB7 23647132 IC50 = 29.6 nM T99041 C60MWC 23647133 IC50 = 126 nM T99041 C8TZD5 23647134 IC50 = 2 nM T99041 CBA8N1 23647136 IC50 = 21 nM T99041 CG0U2M 23647137 IC50 = 33 nM T99041 C3TSN4 23647138 IC50 = 37 nM T99041 C6QKM4 23647139 IC50 = 310 nM T99041 CQPN26 23647141 IC50 = 780 nM T99041 C4V5TC 23647142 IC50 = 995 nM T99041 C8TDA5 23647143 IC50 = 1247 nM T99041 CNRH86 23647144 IC50 = 1325 nM T99041 CY19JV 23647145 IC50 = 1460 nM T99041 C39DJX 23647146 IC50 = 1995 nM T99041 C4P2IJ 23647147 IC50 = 2209 nM T99041 CTB09J 23647311 IC50 = 13 nM T99041 CJ6XT7 23647314 IC50 = 18 nM T99041 CVI19F 23653088 IC50 = 3800 nM T99041 CO9GD8 23655077 IC50 = 22 nM T99041 CWVR37 23655298 IC50 > 500000 nM T99041 CPCX60 23655474 IC50 > 1000000 nM T99041 CB1E5P 23655476 IC50 > 500000 nM T99041 CWTD09 23655478 IC50 > 1000000 nM T99041 CLSE92 23655741 IC50 > 40200 nM T99041 CQ53MU 23655742 IC50 > 36900 nM T99041 C4DOR0 23655937 IC50 > 41300 nM T99041 CRA46X 23655938 IC50 > 39100 nM T99041 CW9UR3 23657402 IC50 > 250000 nM T99041 CU18EA 23657547 IC50 > 250000 nM T99041 CVF6E2 23661697 IC50 = 25 nM T99041 CM7C4W 23661708 IC50 = 26 nM T99041 CO6L9F 23661716 IC50 = 1.2 nM T99041 CHR14F 23661718 IC50 = 6 nM T99041 CG8TJ9 23824719 IC50 = 11000 nM T99041 CNP9T1 24180585 IC50 = 37 nM T99041 CO0ZA3 24692381 IC50 = 67000 nM T99041 CR7I3Y 24703639 IC50 > 1000000 nM T99041 CVA72K 24704198 IC50 = 374000 nM T99041 CKWZ51 24710701 IC50 = 360000 nM T99041 CKVQ51 24749924 IC50 = 1 nM T99041 CCW9N3 24749925 IC50 = 4 nM T99041 CXNY61 24749926 IC50 = 4 nM T99041 CZ4BH0 24749927 IC50 = 284 nM T99041 C9X8CK 24750044 IC50 = 5 nM T99041 CK7V6L 24750165 IC50 = 56 nM T99041 C7I4LK 24750278 IC50 = 3 nM T99041 CT21RV 24750279 IC50 = 2 nM T99041 CC6X1F 24750280 IC50 = 88 nM T99041 C5TIP2 24750281 IC50 = 9 nM T99041 C7QSH2 24752844 IC50 = 65 nM T99041 CI0W8A 24755210 IC50 = 1.3 nM T99041 CU7W4F 24768547 IC50 = 0.21 nM T99041 CX8DH1 24769723 IC50 = 1.4 nM T99041 C0H8OB 24776705 IC50 = 116 nM T99041 C24GLZ 24776939 IC50 = 0.18 nM T99041 C6LD2J 24777439 IC50 = 209 nM T99041 CK8EL5 24777568 IC50 = 12 nM T99041 CQ20PV 24777692 IC50 = 88 nM T99041 C1WF3I 24777804 IC50 = 4.3 nM T99041 C50SPA 24784161 IC50 = 123 nM T99041 C29SZR 24784416 IC50 = 90000 nM T99041 C0H8IZ 24784426 IC50 = 116 nM T99041 CO7L6R 24784427 IC50 = 73 nM T99041 C8FQT4 24784664 IC50 > 100000 nM T99041 C69QMZ 24784674 IC50 = 238 nM T99041 CW8LK2 24784675 IC50 = 47 nM T99041 CH1W5N 24784676 IC50 = 140 nM T99041 CJ0ZI7 24784677 IC50 = 251 nM T99041 CIZF59 24784915 IC50 = 72 nM T99041 CKFH56 24784916 IC50 = 195 nM T99041 C5HY0P 24784918 IC50 = 212 nM T99041 CS6HU2 24784925 IC50 = 182 nM T99041 CK6W8S 24784926 IC50 = 45 nM T99041 CUH32V 24785152 IC50 = 305 nM T99041 C2KL7G 24794725 IC50 = 63 nM T99041 CUM03S 24798754 IC50 = 0.12 nM T99041 CZ3ND1 24832041 IC50 = 32 nM T99041 CY9W8O 24860300 IC50 = 1 nM T99041 CKZ25G 24862861 IC50 = 7.5 nM T99041 CFNZ09 24893980 IC50 = 3670 nM T99041 CMK9B7 24894026 IC50 > 100000 nM T99041 CSIK84 24906298 IC50 = 500000 nM T99041 CYL69J 24951732 IC50 = 0.7 nM T99041 CNP3T1 24951733 IC50 = 3.7 nM T99041 CDCP18 24952087 IC50 = 7.3 nM T99041 CIM7S2 24952089 IC50 = 3.5 nM T99041 CX83WL 24963343 IC50 > 100000 nM T99041 CDU69X 24999325 IC50 = 50 nM T99041 CA94RD 24999327 IC50 = 9 nM T99041 CZJ2N6 24999330 IC50 = 24 nM T99041 C9ML5P 24999630 IC50 = 14 nM T99041 C3VU2K 24999632 IC50 = 69 nM T99041 CUO7Q4 24999636 IC50 = 120 nM T99041 CM6AW8 24999638 IC50 = 39 nM T99041 CY90LJ 25014552 IC50 = 2740 nM T99041 CA28YZ 25017799 IC50 = 2.28 nM T99041 C40ONC 25021195 IC50 = 223 nM T99041 C67ZQD 25054021 IC50 = 357 nM T99041 C3SW1V 25054553 IC50 = 64 nM T99041 CH9F2B 25054555 IC50 = 64 nM T99041 CHO68D 25054557 IC50 = 56 nM T99041 C3R9XM 25054809 IC50 = 50 nM T99041 C2D4LI 25054811 IC50 = 3 nM T99041 CHE83A 25054815 IC50 = 13 nM T99041 CXPO63 25054817 IC50 = 68 nM T99041 CA2EK8 25055067 IC50 = 328 nM T99041 C8J9ZG 25055304 IC50 = 80 nM T99041 C51KTQ 25055741 IC50 = 7.4 nM T99041 CI0K2T 25055743 IC50 = 4.3 nM T99041 C1Q6RS 25055745 IC50 = 2.2 nM T99041 CIA48J 25055828 IC50 = 204 nM T99041 CA3N5B 25055836 IC50 = 229 nM T99041 CEDP80 25055999 IC50 = 1.7 nM T99041 C5K3QM 25056001 IC50 = 11 nM T99041 CGX3K8 25056003 IC50 = 17 nM T99041 C6X9PG 25056005 IC50 = 5.2 nM T99041 C8P7VJ 25056091 IC50 = 601 nM T99041 CN83UK 25056093 IC50 = 77 nM T99041 C0LJF5 25056353 IC50 = 6 nM T99041 CS81DK 25056618 IC50 = 112 nM T99041 CQM3U1 25056620 IC50 = 192 nM T99041 C7WEY3 25056875 IC50 = 807 nM T99041 C62UCV 25056881 IC50 = 95 nM T99041 CK7B2E 25057130 IC50 = 102 nM T99041 CQCY54 25057136 IC50 = 25 nM T99041 CM3AU5 25057138 IC50 = 17 nM T99041 CR26DS 25057390 IC50 = 309 nM T99041 C8Q2GP 25057392 IC50 = 175 nM T99041 C9TQ7J 25057396 IC50 = 680 nM T99041 C6KHT4 25057400 IC50 = 1700 nM T99041 C6Q2CM 25057648 IC50 = 88 nM T99041 C1RN5F 25057650 IC50 = 101 nM T99041 CUF2P9 25057652 IC50 = 212 nM T99041 CQHM69 25110577 IC50 = 510 nM T99041 CTS7I5 25110685 IC50 = 3.6 nM T99041 CHTM74 25110898 IC50 = 2500 nM T99041 CBC24W 25110901 IC50 = 8500 nM T99041 CW3GZ6 25112031 IC50 = 710 nM T99041 C76RFD 25112033 IC50 = 2200 nM T99041 CYV1T4 25112035 IC50 = 1900 nM T99041 CW7UD1 25112037 IC50 = 1600 nM T99041 CX9NR5 25112039 IC50 = 3000 nM T99041 CN2MQ8 25112155 IC50 = 770 nM T99041 CO7UE8 25112157 IC50 = 3700 nM T99041 CUIW48 25112159 IC50 = 3100 nM T99041 C6B8CF 25112161 IC50 = 2000 nM T99041 CQ0GY8 25112163 IC50 = 1600 nM T99041 CI71VQ 25112265 IC50 = 8900 nM T99041 CR13HD 25112267 IC50 = 1900 nM T99041 CWE10R 25112269 IC50 = 3600 nM T99041 CK69WG 25112271 IC50 = 1400 nM T99041 C5W8KL 25112273 IC50 = 5900 nM T99041 CXM0N5 25112374 IC50 = 2800 nM T99041 CK16JS 25112376 IC50 = 4300 nM T99041 C9KF5T 25112378 IC50 = 2200 nM T99041 C5O9PU 25112380 IC50 = 2700 nM T99041 C19DPQ 25112382 IC50 = 1400 nM T99041 CYJ2B5 25112487 IC50 = 2700 nM T99041 CUA2K9 25112489 IC50 = 1600 nM T99041 C60EOS 25112491 IC50 = 5600 nM T99041 CV75BU 25112493 IC50 = 1600 nM T99041 CDL2S7 25112495 IC50 = 7400 nM T99041 CF97YP 25112497 IC50 = 1300 nM T99041 CDKE79 25112619 IC50 = 2100 nM T99041 C4TLZ7 25112621 IC50 = 9100 nM T99041 CI3KP5 25112623 IC50 = 690 nM T99041 CF9BO5 25112625 IC50 = 4800 nM T99041 C5QA1K 25112627 IC50 = 2600 nM T99041 C01GPL 25132159 Ki = 8.3 nM T99041 C7IDX9 25132160 IC50 = 0.89 nM T99041 C9VK8W 25132161 Ki = 17 nM T99041 CFZ4V2 25132162 Ki = 3300 nM T99041 CSU0B5 25189891 Ki = 14.4 nM T99041 CA98HO 25203967 IC50 = 2000 nM T99041 CPMN48 28787393 IC50 = 6.29 nM T99041 C9Q2OH 42601533 IC50 = 3850 nM T99041 C0BC9N 42601535 IC50 = 350 nM T99041 C7KN2U 42608447 IC50 = 0.38 nM T99041 C60SVD 42636924 IC50 = 15 nM T99041 C76NLT 42773972 IC50 > 250000 nM T99041 C6LQN3 43181622 IC50 > 1000000 nM T99041 C42OZD 43271345 IC50 = 377000 nM T99041 CK54OM 43650152 IC50 = 229000 nM T99041 CS40ML 44123747 IC50 = 1.1 nM T99041 CSX10M 44138030 IC50 = 4 nM T99041 CQF86D 44182505 IC50 = 13 nM T99041 C3I4TF 44201003 IC50 = 10 nM T99041 CE5B7H 44218404 IC50 = 13 nM T99041 CR8GT4 44218550 IC50 = 15 nM T99041 CBW7D4 44218551 IC50 = 39 nM T99041 CVH08B 44218552 IC50 = 18 nM T99041 CISE95 44218553 IC50 = 27 nM T99041 CLB72R 44218554 IC50 = 14 nM T99041 C2N9VR 44218555 IC50 = 63 nM T99041 CJ6L3S 44218693 IC50 = 29 nM T99041 C97IFE 44218695 IC50 = 32 nM T99041 C50EKW 44250174 IC50 = 9 nM T99041 CRZI12 44266022 IC50 = 14 nM T99041 C9YT6M 44270944 Ki = 1.1 nM T99041 C4MSN1 44285301 IC50 = 7900 nM T99041 CP9YN0 44285888 IC50 = 7000 nM T99041 CT3U1W 44286225 IC50 = 2400 nM T99041 C5UA6S 44286288 IC50 = 103000 nM T99041 CMG71F 44286291 IC50 = 52600 nM T99041 CQ5H8W 44286293 IC50 = 18000 nM T99041 CB6R9L 44286310 IC50 = 948000 nM T99041 C7ZHL3 44286477 IC50 = 277000 nM T99041 CF2H7C 44286480 IC50 = 746000 nM T99041 C7YU4C 44286501 IC50 = 6700 nM T99041 C0HZ5A 44286513 IC50 = 8400 nM T99041 C54LIM 44286562 IC50 = 170000 nM T99041 CH72YN 44286743 IC50 = 31800 nM T99041 C58LKI 44286823 IC50 = 14000 nM T99041 CVQ7K3 44286825 IC50 = 4700 nM T99041 CL3Q2J 44306072 IC50 = 4000 nM T99041 CMC8B9 44306777 IC50 = 44 nM T99041 CF2Q5V 44325514 Ki = 0.5 nM T99041 CE6G4X 44325523 Ki = 450 nM T99041 CI2YN1 44325525 Ki = 260 nM T99041 C29OIF 44325533 Ki = 0.8 nM T99041 CV4QM7 44325534 Ki = 6000 nM T99041 CLDY18 44325535 Ki = 4200 nM T99041 CN46PE 44325540 Ki = 21 nM T99041 CX94HW 44325697 Ki = 5 nM T99041 C1GRJ2 44325719 Ki = 0.41 nM T99041 CN45KP 44325734 Ki = 1.7 nM T99041 C4WTQ7 44326630 IC50 = 109000 nM T99041 C98LVO 44326651 IC50 = 372 nM T99041 C51EOL 44326652 IC50 = 218 nM T99041 C49PEQ 44326772 IC50 = 18700 nM T99041 C8NS4L 44326791 IC50 = 242 nM T99041 CYHE81 44327018 IC50 = 256 nM T99041 CNH8J3 44327071 IC50 = 16 nM T99041 CR3GE1 44327072 IC50 = 15 nM T99041 CSU32T 44327098 IC50 = 377 nM T99041 C0XFT4 44327160 IC50 = 13 nM T99041 CG7K1P 44327192 IC50 = 123 nM T99041 C2RC9I 44328126 IC50 = 14000 nM T99041 CTC40N 44328274 Ki = 47600 nM T99041 C8M0SH 44328300 Ki = 200 nM T99041 C6NZ9C 44328318 IC50 = 213000 nM T99041 C6OHV2 44328319 IC50 > 500000 nM T99041 CA53DN 44330624 IC50 = 13000 nM T99041 C7E1BJ 44330636 IC50 = 68000 nM T99041 C75JRD 44360575 IC50 = 24 nM T99041 CS72FI 44360697 IC50 = 7.5 nM T99041 CKSO92 44360724 IC50 = 26 nM T99041 CYED53 44360725 IC50 = 89 nM T99041 CXEC92 44360726 IC50 = 35 nM T99041 CL7WM8 44360734 IC50 = 64 nM T99041 CA0U8X 44360744 IC50 = 98 nM T99041 C50NME 44360749 IC50 = 94 nM T99041 CKI6W3 44360785 IC50 = 18 nM T99041 CRM9Y7 44360786 IC50 = 24 nM T99041 CXTP74 44360787 IC50 = 2.6 nM T99041 C5MB1D 44360809 IC50 = 46 nM T99041 C29DTA 44360810 IC50 = 190 nM T99041 CPTX82 44360812 IC50 = 2700 nM T99041 C3M8KF 44360910 IC50 = 38 nM T99041 CR7Q9N 44360911 IC50 = 53 nM T99041 CFY7P3 44360924 IC50 = 33 nM T99041 C62HNE 44360925 IC50 = 33 nM T99041 C1H5YG 44360938 IC50 = 21 nM T99041 C6IZ8L 44360955 IC50 = 15 nM T99041 CCJA09 44360967 IC50 = 29 nM T99041 CLMF32 44360976 IC50 = 20 nM T99041 CV1YL5 44360977 IC50 = 17 nM T99041 CY8A9K 44361010 IC50 = 10 nM T99041 C2KWI0 44361074 IC50 = 17 nM T99041 C1Z2FV 44361086 IC50 = 55 nM T99041 C8MJY5 44361216 IC50 = 9 nM T99041 CYK42S 44361230 IC50 = 25 nM T99041 CM3R2T 44364102 IC50 = 250000 nM T99041 CJ0VM6 44364126 IC50 = 3500 nM T99041 C83IUZ 44364133 IC50 = 217000 nM T99041 CJ8N0S 44364172 IC50 > 1000000 nM T99041 C7D2FW 44364210 IC50 = 93000 nM T99041 C8HO2F 44364211 IC50 = 500000 nM T99041 C9IQG4 44364212 IC50 > 1000000 nM T99041 C47NKP 44364213 IC50 = 52000 nM T99041 C6CYU9 44364227 IC50 > 500000 nM T99041 CHLV59 44364231 IC50 > 500000 nM T99041 CZF5N2 44364237 IC50 > 1000000 nM T99041 C7VR0N 44364252 IC50 > 1000000 nM T99041 CTS8U3 44364253 IC50 > 1000000 nM T99041 C0IW9L 44364296 IC50 = 289000 nM T99041 C6FBH7 44364297 IC50 = 81000 nM T99041 C79JMS 44364298 IC50 = 318000 nM T99041 CF2TA0 44364385 IC50 = 151000 nM T99041 C19DCN 44364405 IC50 = 51000 nM T99041 CX5AK7 44364446 IC50 > 500000 nM T99041 C4XIV2 44364456 IC50 > 1000000 nM T99041 C3XN5A 44364457 IC50 = 107000 nM T99041 CKA86J 44364458 IC50 = 500000 nM T99041 C4QON9 44368427 IC50 = 12.8 ug.mL-1 T99041 C8FB1S 44368725 IC50 = 64.4 ug.mL-1 T99041 CE83AK 44368726 IC50 > 100 ug.mL-1 T99041 CW9BG0 44368735 IC50 = 18.7 ug.mL-1 T99041 C37TIM 44368736 IC50 = 15.1 ug.mL-1 T99041 CX8I6C 44381633 IC50 = 550 nM T99041 CW9F3N 44381634 IC50 = 1200 nM T99041 CI39RJ 44381635 IC50 = 210 nM T99041 CLK90J 44381645 IC50 = 95 nM T99041 CT0EO4 44381646 IC50 = 240 nM T99041 CHX2T7 44381647 IC50 = 1100 nM T99041 C6Y4QW 44381687 IC50 = 110 nM T99041 CN96MI 44381721 IC50 = 420 nM T99041 CK4SP1 44381763 IC50 = 480 nM T99041 CI6RT5 44381811 IC50 = 4600 nM T99041 CG1CD7 44381826 IC50 = 110 nM T99041 CL51SX 44381845 IC50 = 660 nM T99041 CXBY42 44381846 IC50 = 230 nM T99041 C5SV9U 44381847 IC50 = 110 nM T99041 CRY5K1 44381848 IC50 = 3900 nM T99041 CRE8J7 44381849 IC50 = 280 nM T99041 CUX2Q9 44381861 IC50 = 220 nM T99041 C92CKY 44381862 IC50 = 130 nM T99041 CIX09S 44381884 IC50 = 46 nM T99041 C3GH0S 44381896 IC50 = 43 nM T99041 C0FQO1 44381899 IC50 = 47 nM T99041 CTRX81 44381910 IC50 = 420 nM T99041 C2XBA5 44381911 IC50 = 170 nM T99041 CBL60E 44381919 IC50 = 250 nM T99041 CARK25 44381928 IC50 = 94 nM T99041 C4LR3K 44381945 IC50 = 270 nM T99041 CQ4VZ3 44381966 IC50 = 440 nM T99041 CDCY49 44381967 IC50 = 670 nM T99041 CT9IN5 44381974 IC50 = 330 nM T99041 C0FQY4 44381979 IC50 = 180 nM T99041 CP7XG9 44382005 IC50 = 180 nM T99041 C6YFP9 44382006 IC50 = 870 nM T99041 CWJ3V5 44382013 IC50 = 1700 nM T99041 CI8O3F 44382065 IC50 = 150 nM T99041 CX2JS7 44382077 IC50 = 72 nM T99041 C38MSH 44382133 IC50 = 110 nM T99041 C8PD7J 44382134 IC50 = 83 nM T99041 C89LXF 44382393 IC50 = 840 nM T99041 CAJ50V 44382443 IC50 = 290 nM T99041 C8ZP1A 44382444 IC50 = 110 nM T99041 CKOD04 44382521 IC50 = 83 nM T99041 CY2C8J 44387751 IC50 > 1000000 nM T99041 CXSU53 44387755 IC50 > 1000000 nM T99041 CALG81 44387756 IC50 > 1000000 nM T99041 CL1M7V 44387758 IC50 > 125000 nM T99041 C6T2MW 44387765 IC50 > 1000000 nM T99041 CA7KI2 44390794 IC50 = 13000 nM T99041 CVD21W 44393563 IC50 = 39640 nM T99041 C24PMT 44393585 IC50 > 100000 nM T99041 CB9WA5 44393586 IC50 = 16480 nM T99041 C7N1GB 44393611 IC50 = 3000 nM T99041 CS51KL 44393656 IC50 = 33000 nM T99041 C7SB1I 44393657 IC50 = 44860 nM T99041 C9JT0N 44393695 IC50 = 46910 nM T99041 CPG38C 44393696 IC50 = 27470 nM T99041 CF6KR8 44393727 IC50 = 51000 nM T99041 C58KPC 44393728 IC50 = 5700 nM T99041 CDH6J1 44393857 IC50 = 200 nM T99041 C2PK9W 44393881 IC50 = 2620 nM T99041 CB6E5I 44393933 IC50 = 80 nM T99041 C08BMZ 44394001 IC50 = 51 nM T99041 C8RA0W 44394023 IC50 = 9400 nM T99041 C3KH1Q 44394024 IC50 = 589 nM T99041 C4QE5X 44394028 IC50 = 143 nM T99041 CPF49E 44394029 IC50 = 155 nM T99041 C8ZA9M 44394031 IC50 = 11000 nM T99041 CS35UP 44394072 IC50 = 2026 nM T99041 CW79MD 44394073 IC50 = 19 nM T99041 CW81MP 44394103 IC50 = 270 nM T99041 C7Y4LZ 44394104 IC50 = 8476 nM T99041 C25SDY 44394118 IC50 = 19000 nM T99041 CU85FA 44394119 IC50 = 30 nM T99041 CJ18AZ 44394135 IC50 = 35000 nM T99041 CTEP50 44394136 IC50 = 36000 nM T99041 C4BO3S 44394155 IC50 = 34 nM T99041 CALF89 44394157 IC50 = 0.1 nM T99041 C4B9OH 44394173 IC50 = 1100 nM T99041 CX75VF 44394180 IC50 = 14860 nM T99041 C85SEO 44394194 IC50 = 2519 nM T99041 CS1Z7X 44394195 IC50 = 2263 nM T99041 C39LZT 44394203 IC50 = 3028 nM T99041 CF6Y8L 44394209 IC50 = 10700 nM T99041 CQ09FB 44394210 IC50 = 1040 nM T99041 CXG8B6 44394238 IC50 = 931 nM T99041 CIJ95E 44394239 IC50 = 981 nM T99041 C3Q5WZ 44394241 IC50 = 3611 nM T99041 CL3EP4 44394242 IC50 = 690 nM T99041 C8U2ZQ 44394244 IC50 = 3279 nM T99041 CZA46H 44394270 IC50 = 2026 nM T99041 CUGH58 44394271 IC50 = 8951 nM T99041 CU7PY3 44394282 IC50 = 7688 nM T99041 C41ITO 44394305 IC50 = 1900 nM T99041 CG53YO 44394349 IC50 = 1552 nM T99041 C59NLA 44394350 IC50 = 1700 nM T99041 C0NSL3 44396153 IC50 = 4 nM T99041 C1VLP6 44399148 IC50 = 252 nM T99041 CIED90 44399244 IC50 = 87 nM T99041 C3PKV8 44399546 IC50 = 97 nM T99041 CEW52I 44400445 IC50 = 0.25 nM T99041 C8UDI1 44400447 IC50 = 0.33 nM T99041 CZ19WH 44400450 IC50 = 6.6 nM T99041 C0MEB2 44400462 IC50 = 1.5 nM T99041 C41SZA 44400473 IC50 = 0.28 nM T99041 C68USM 44400485 IC50 = 0.19 nM T99041 CZ6A8Q 44400504 IC50 = 3 nM T99041 CJD9B5 44400535 IC50 = 5.5 nM T99041 CU8CL1 44400547 IC50 = 6.7 nM T99041 CR87KM 44400555 IC50 = 1.9 nM T99041 CSJU72 44400574 IC50 = 4.6 nM T99041 C6VB2Q 44400588 IC50 = 9.7 nM T99041 C3RAW7 44400625 IC50 = 0.53 nM T99041 CUR51H 44402967 Ki = 504 nM T99041 CZO5J3 44402970 Ki = 1267 nM T99041 CIKW98 44402971 Ki = 61 nM T99041 CP72TO 44402972 Ki = 81 nM T99041 CA8K9B 44403068 Ki = 109 nM T99041 C32LIY 44403069 Ki = 117 nM T99041 CPX1M9 44403336 IC50 = 370 nM T99041 CSEN70 44403337 IC50 = 17000 nM T99041 C0NXE8 44403338 IC50 = 2000 nM T99041 CR53EK 44403354 IC50 = 1200 nM T99041 CRO16Q 44403360 IC50 = 4.5 nM T99041 C0FC7D 44403361 IC50 = 15 nM T99041 C3HFZ7 44403391 IC50 = 130 nM T99041 C3TOY4 44403392 IC50 = 75 nM T99041 CU39LX 44403393 IC50 = 25 nM T99041 CIA8Y3 44403397 IC50 = 27 nM T99041 C6P7NE 44403398 IC50 = 58 nM T99041 CP34SF 44403405 IC50 = 8 nM T99041 C60VBT 44403406 IC50 = 61 nM T99041 C50LWV 44403411 IC50 = 16000 nM T99041 CQ5T4Y 44403412 IC50 = 0.8 nM T99041 CMX9B1 44403416 IC50 = 12 nM T99041 CUKG07 44403417 IC50 = 560 nM T99041 CX29FU 44403421 IC50 = 1600 nM T99041 C2P4CQ 44403422 IC50 = 7.8 nM T99041 CCOA39 44403438 IC50 = 32000 nM T99041 CLYJ80 44403439 IC50 = 810 nM T99041 C4YAH3 44404393 IC50 = 25 nM T99041 C02SYC 44406179 Ki = 225 nM T99041 CU8B3S 44406189 Ki = 46 nM T99041 C1SBD5 44406234 Ki = 115 nM T99041 C5P1RX 44406284 Ki = 40 nM T99041 C0IQO3 44411572 IC50 = 771 nM T99041 C3HXA1 44411573 IC50 > 3000 nM T99041 CW73SO 44411579 IC50 > 3000 nM T99041 CB17FI 44411652 IC50 > 3000 nM T99041 C5WPL4 44411659 IC50 > 3000 nM T99041 C1HCZ6 44411660 IC50 > 3000 nM T99041 C29ZOU 44411665 IC50 > 3000 nM T99041 C9MH4X 44411669 IC50 > 3000 nM T99041 C54RFY 44411670 IC50 > 3000 nM T99041 CE86UP 44411700 IC50 = 237 nM T99041 CR7MX8 44411923 IC50 = 1860 nM T99041 CFP80H 44412105 Ki = 0.41 nM T99041 CZ15VN 44412163 Ki = 2.5 nM T99041 C0HA7I 44412169 Ki = 2900 nM T99041 CGJ17L 44415883 IC50 > 250000 nM T99041 CE0KW2 44415905 IC50 > 100000 nM T99041 CPR49A 44415906 IC50 > 125000 nM T99041 CQ5P2J 44415929 IC50 = 234000 nM T99041 CM2W5X 44415930 IC50 > 125000 nM T99041 COPZ87 44415944 IC50 > 125000 nM T99041 CGLB32 44417381 Ki = 49 nM T99041 C2TP5K 44417385 Ki = 97 nM T99041 CN2F6U 44417389 Ki > 30000 nM T99041 C12HGD 44417391 Ki > 30000 nM T99041 CSG4F8 44417393 Ki = 1 nM T99041 CE7UB0 44418114 IC50 = 0.29 nM T99041 CD9J3S 44418157 IC50 = 4 nM T99041 C70KAO 44418211 IC50 = 42 nM T99041 C8LC2A 44418213 IC50 = 127 nM T99041 CTM1Y8 44418214 IC50 = 269 nM T99041 C1EMA5 44418215 IC50 = 144 nM T99041 CWDH12 44418216 IC50 = 1300 nM T99041 C1FB4K 44418218 IC50 = 252 nM T99041 CVC3R4 44418219 IC50 = 236 nM T99041 CU1FG2 44418222 IC50 = 247 nM T99041 C8ZH5R 44418223 IC50 = 320 nM T99041 CA9YM3 44418225 IC50 = 232 nM T99041 CQE5Y0 44418229 IC50 = 181 nM T99041 CID62U 44418230 Ki = 4300 nM T99041 CI2H7Q 44418231 Ki = 9080 nM T99041 C2LXS7 44418232 IC50 = 118 nM T99041 CXCV19 44418233 Ki = 7391 nM T99041 CZW38C 44418239 Ki = 9500 nM T99041 C7KF0X 44418240 Ki = 4600 nM T99041 C8QJ7H 44418242 Ki = 19500 nM T99041 C60KPZ 44418243 Ki = 11300 nM T99041 CMKW39 44418246 Ki = 68 nM T99041 CEBQ24 44418249 Ki = 1430 nM T99041 C59HZQ 44418251 IC50 = 8000 nM T99041 CDX2Q5 44418253 Ki = 451000 nM T99041 C0RV8O 44418254 Ki = 182000 nM T99041 C37KEO 44418255 Ki = 6871 nM T99041 C2UR9X 44418256 IC50 = 239 nM T99041 CK20CA 44418257 IC50 = 190 nM T99041 CO3GL6 44418260 IC50 = 207 nM T99041 CY3O7C 44418261 IC50 = 197 nM T99041 C0ITV9 44418262 IC50 = 433 nM T99041 CGR3H7 44418263 IC50 = 21000 nM T99041 C68SHD 44418264 IC50 = 253 nM T99041 CDI98V 44418265 IC50 = 225 nM T99041 CHO5P1 44418266 IC50 = 911 nM T99041 C95XQC 44418268 IC50 = 174 nM T99041 CE3C4D 44420996 Ki = 140 nM T99041 CI2P6M 44420998 Ki = 6.1 nM T99041 C0FT8Q 44420999 Ki = 4 nM T99041 C7VU1I 44421000 Ki = 13 nM T99041 C38PJE 44421001 Ki = 2.3 nM T99041 CX4C3Y 44421002 Ki = 11 nM T99041 CF52AI 44421003 Ki = 23 nM T99041 C6NV0S 44421004 Ki = 1.6 nM T99041 C5W8VX 44421005 Ki = 2.3 nM T99041 C8KC3R 44421006 Ki = 3 nM T99041 C16YHQ 44422417 IC50 = 112 nM T99041 C9IRG5 44422418 IC50 = 11 nM T99041 C7XU0J 44422419 IC50 = 7.9 nM T99041 C58WCU 44422439 IC50 = 19.2 nM T99041 C2F9DG 44422440 IC50 = 51.5 nM T99041 CS63GZ 44422443 IC50 = 5.8 nM T99041 C9M5YC 44422444 IC50 = 7 nM T99041 C0J1UX 44422445 IC50 = 45.4 nM T99041 CKFM17 44422448 IC50 = 6.5 nM T99041 C6C3ZF 44422475 IC50 = 147 nM T99041 C9T1KM 44422476 IC50 = 25.2 nM T99041 CN5G6O 44422477 IC50 = 181 nM T99041 CNQC83 44422485 IC50 = 34 nM T99041 C5NK2E 44422486 IC50 > 300 nM T99041 CZ5UW9 44422487 IC50 = 37.2 nM T99041 C6TZM8 44422496 IC50 > 300 nM T99041 CX5M3Q 44422497 IC50 > 300 nM T99041 C86SXN 44422498 IC50 = 154 nM T99041 C4YP0T 44422507 IC50 = 85.9 nM T99041 C1IW2L 44422508 IC50 > 300 nM T99041 CRWM46 44422509 IC50 > 300 nM T99041 CJK1H2 44422513 IC50 = 9.6 nM T99041 C6C5PM 44422514 IC50 = 7.1 nM T99041 C4KSW0 44422518 IC50 = 9.1 nM T99041 CL40CD 44422519 IC50 = 6.4 nM T99041 CY4K6X 44422522 IC50 = 13.6 nM T99041 CZ8TO9 44422523 IC50 = 13.9 nM T99041 CCFT17 44422525 IC50 = 16.8 nM T99041 C0BXJ2 44422526 IC50 = 17 nM T99041 CGB32F 44422527 IC50 = 228 nM T99041 C1N4RA 44422528 IC50 = 26.4 nM T99041 C1D7ER 44425490 IC50 = 8 nM T99041 CZ2MB8 44426068 IC50 = 6.6 nM T99041 C8PKO5 44426070 IC50 = 139 nM T99041 CW7QD8 44429116 IC50 = 3.5 nM T99041 C1NF6D 44429117 IC50 = 3.4 nM T99041 CG67NO 44429119 IC50 = 5.7 nM T99041 CT54EH 44429120 IC50 = 2.9 nM T99041 C37SUV 44429122 IC50 = 2.4 nM T99041 C57GUJ 44429124 IC50 = 7.8 nM T99041 CW59YC 44429127 IC50 = 3.5 nM T99041 C0L9SG 44429129 IC50 = 6.1 nM T99041 CT2P8M 44429130 IC50 = 9.1 nM T99041 C4KRA5 44429131 IC50 = 3.9 nM T99041 CM2FK3 44429132 IC50 = 2.5 nM T99041 CEL8D9 44429133 IC50 = 3.3 nM T99041 CX48BO 44429134 IC50 = 8.3 nM T99041 CWF04T 44429135 IC50 = 23 nM T99041 CN68CG 44429136 IC50 = 8.9 nM T99041 C6J3CS 44429137 IC50 = 22 nM T99041 C6F1NE 44429138 IC50 = 4.9 nM T99041 CL2G7Z 44429139 IC50 = 7.1 nM T99041 CHT96Z 44429140 IC50 = 5.3 nM T99041 CVD9U0 44429602 IC50 = 3.8 nM T99041 C17MKX 44429603 IC50 = 16 nM T99041 C3SKR2 44429609 IC50 = 4.5 nM T99041 C0SU2X 44429610 IC50 = 2.4 nM T99041 CGQN20 44429612 IC50 = 7.7 nM T99041 CYGD28 44429613 IC50 = 3.5 nM T99041 CZ7LW9 44429614 IC50 = 4.4 nM T99041 CXJD74 44429616 IC50 = 5.7 nM T99041 C6R2IZ 44429619 IC50 = 6 nM T99041 C0A2CF 44429620 IC50 = 4 nM T99041 C4EH0L 44429622 IC50 = 4.9 nM T99041 CY4MF9 44429623 IC50 = 8.3 nM T99041 C02JQU 44429624 IC50 = 11 nM T99041 CG3C7E 44429625 IC50 = 4.3 nM T99041 CHNV25 44429626 IC50 = 4.8 nM T99041 C7IL3S 44431164 IC50 = 98 nM T99041 C0UOS8 44431165 IC50 = 135 nM T99041 CEG05S 44431166 IC50 = 272 nM T99041 CO8S3Z 44431170 IC50 = 805 nM T99041 C2K4RQ 44431176 IC50 = 151 nM T99041 CJZY21 44431177 IC50 = 87 nM T99041 CSJI40 44431185 IC50 = 1018 nM T99041 C36EJR 44431188 IC50 = 486 nM T99041 C2MCA1 44431191 IC50 = 366 nM T99041 C89XVB 44431197 IC50 = 511 nM T99041 CK76EP 44431199 IC50 = 145 nM T99041 C3FPT2 44431200 IC50 = 59 nM T99041 C4F8AG 44431201 IC50 = 264 nM T99041 CWX4I3 44431203 IC50 = 1580 nM T99041 CZ3N9E 44431204 IC50 = 23 nM T99041 C5NAS6 44431205 IC50 = 180 nM T99041 C37SGU 44431206 IC50 = 84 nM T99041 CYD62G 44431212 IC50 = 60 nM T99041 C72WTP 44431213 IC50 = 30 nM T99041 CC3T9G 44431214 IC50 = 65 nM T99041 CL4T3X 44431215 IC50 = 190 nM T99041 C4WVL8 44431216 IC50 = 69 nM T99041 CO08HZ 44431217 IC50 = 37 nM T99041 CCPZ23 44431218 IC50 = 30 nM T99041 C0J7WV 44431219 IC50 = 29 nM T99041 C16ZTV 44431220 IC50 = 219 nM T99041 CR0A1M 44431316 IC50 = 21 nM T99041 CV1R7A 44431317 IC50 = 140 nM T99041 CTB82G 44431744 IC50 = 520 nM T99041 C7O4GL 44431746 IC50 = 35700 nM T99041 CJOR92 44431752 IC50 = 2100 nM T99041 CETI27 44431756 IC50 = 5800 nM T99041 C2VY9T 44431757 IC50 = 142000 nM T99041 C09BFG 44431758 IC50 = 2600 nM T99041 CX3ZH1 44431759 IC50 = 4900 nM T99041 C5JYG0 44431760 IC50 = 26000 nM T99041 C1CRX9 44431761 IC50 = 2300 nM T99041 CB7SA0 44431762 IC50 = 18400 nM T99041 C4FT0P 44431764 IC50 = 8900 nM T99041 C7OJW0 44431765 IC50 = 220 nM T99041 CMU40B 44431766 IC50 = 990 nM T99041 CA9P1R 44431767 IC50 = 1520 nM T99041 CL0VB1 44431768 IC50 = 10590 nM T99041 CHG8I4 44431769 IC50 = 370 nM T99041 C7PLH0 44431770 IC50 = 9380 nM T99041 CC0J6A 44431771 IC50 = 3730 nM T99041 C4X1GA 44431772 IC50 = 5130 nM T99041 C4S8DE 44431773 IC50 = 650 nM T99041 CQX2S0 44431774 IC50 = 32 nM T99041 CL6B7S 44431775 IC50 = 4 nM T99041 C16CRQ 44431776 IC50 = 50 nM T99041 CY76AB 44432858 IC50 = 77 nM T99041 CS95EU 44432859 IC50 = 67 nM T99041 C1PX9V 44432860 IC50 = 223 nM T99041 C3AN4E 44432861 IC50 = 7939 nM T99041 CE4Q5X 44432862 IC50 = 35 nM T99041 CHN6E3 44432863 IC50 = 63 nM T99041 CF2AT6 44432881 IC50 = 15 nM T99041 CTD24F 44432889 IC50 = 95 nM T99041 CSC2E0 44432894 IC50 = 210 nM T99041 CU67PL 44432901 IC50 = 224 nM T99041 C35GZP 44432904 IC50 = 84 nM T99041 C21UQD 44432911 IC50 = 53 nM T99041 CU27DF 44432914 IC50 = 680 nM T99041 C9E1SZ 44432915 IC50 = 339 nM T99041 CZ47KB 44432929 IC50 = 20 nM T99041 CS5BT9 44432935 IC50 = 56 nM T99041 CI9M8R 44432936 IC50 = 17 nM T99041 C5LTR0 44432937 IC50 = 30 nM T99041 C6EJB0 44432938 IC50 = 10 nM T99041 CJ7YN0 44432940 IC50 = 255 nM T99041 CVZ3I2 44432942 IC50 = 47 nM T99041 CT29BC 44432944 IC50 = 25 nM T99041 CNOW68 44433160 IC50 = 140 nM T99041 CJUH82 44433161 IC50 = 2000 nM T99041 C8A1ZL 44433162 IC50 = 150 nM T99041 CJ61CN 44433163 IC50 > 3000 nM T99041 C20OBQ 44433164 IC50 > 3000 nM T99041 C1GBW2 44433165 IC50 > 3000 nM T99041 CEJC97 44433166 IC50 > 3000 nM T99041 CI1NU4 44433167 IC50 = 1000 nM T99041 C5NAI2 44433168 IC50 > 3000 nM T99041 C7TWF9 44433169 IC50 > 3000 nM T99041 C5YUC3 44433174 Ki = 1420 nM T99041 CI5UK4 44433203 IC50 = 790 nM T99041 CVL2Q7 44433204 IC50 = 1400 nM T99041 CR5X3V 44433205 IC50 = 2300 nM T99041 CGB9I5 44433206 IC50 = 2900 nM T99041 CZGM71 44433207 IC50 > 3000 nM T99041 C8PBJ4 44433208 IC50 > 3000 nM T99041 CQ71FG 44433209 IC50 > 3000 nM T99041 C3QOB8 44433210 IC50 > 3000 nM T99041 CO8WI2 44433212 IC50 > 3000 nM T99041 COC75P 44433213 IC50 > 3000 nM T99041 CIB5K2 44433214 IC50 > 3000 nM T99041 C7LI5A 44433215 IC50 > 3000 nM T99041 CCT2I4 44433216 IC50 = 260 nM T99041 CTA59M 44433217 IC50 = 93 nM T99041 CY73TI 44433218 IC50 = 230 nM T99041 C91CFD 44433219 IC50 = 57 nM T99041 CAN07M 44433220 IC50 = 180 nM T99041 C4UTL0 44433221 IC50 = 190 nM T99041 C8CWB2 44433222 IC50 = 37 nM T99041 C4O8SB 44433223 IC50 = 19 nM T99041 CQDS95 44433224 IC50 = 14 nM T99041 CNW1S2 44433225 IC50 = 47 nM T99041 CB04FG 44433226 IC50 = 470 nM T99041 C90GFZ 44433227 IC50 = 130 nM T99041 CSHA84 44433228 IC50 = 160 nM T99041 C6ZP3F 44433229 IC50 = 51 nM T99041 C7KR9C 44433230 IC50 = 120 nM T99041 CH96JN 44433231 IC50 = 71 nM T99041 CR7CQ3 44433232 IC50 = 1300 nM T99041 CWI98S 44433233 IC50 = 32 nM T99041 C23ZRQ 44433234 IC50 = 14 nM T99041 C43RDG 44433235 IC50 = 120 nM T99041 CU6O4S 44433236 IC50 = 70 nM T99041 C8U4QI 44433237 IC50 = 31 nM T99041 C9GIE3 44433617 IC50 = 16 nM T99041 C5B4HS 44433618 IC50 = 12 nM T99041 CU6XZ5 44433646 IC50 = 100 nM T99041 CM8E2D 44433661 IC50 = 38 nM T99041 C07PZD 44433929 Ki > 10000 nM T99041 CG8QR0 44433931 Ki = 3653 nM T99041 CMG6W7 44433932 Ki = 877 nM T99041 CMUR94 44433933 Ki > 10000 nM T99041 CU7AR9 44433934 Ki = 3007 nM T99041 C1ML6S 44433935 Ki > 10000 nM T99041 CM9V3B 44433936 Ki > 10000 nM T99041 C0PLN8 44433937 Ki > 10000 nM T99041 CE5F7Q 44433938 Ki > 10000 nM T99041 CCBR97 44433939 Ki > 10000 nM T99041 CCEO15 44433941 Ki > 10000 nM T99041 CL6V0G 44433942 Ki > 10000 nM T99041 CB70WG 44433943 Ki > 10000 nM T99041 CC02JQ 44433944 Ki > 10000 nM T99041 C9SO3Y 44433945 Ki = 3257 nM T99041 CU7WB6 44433946 Ki > 10000 nM T99041 CAD8G1 44433950 Ki = 1010 nM T99041 C1P2BE 44433951 Ki = 1065 nM T99041 CZA08G 44433952 Ki = 530 nM T99041 CIJF53 44433953 Ki = 731 nM T99041 CTF97G 44433954 Ki = 356 nM T99041 CQ9JD6 44433955 Ki > 10000 nM T99041 CP0M9W 44433956 Ki > 10000 nM T99041 CQ41OU 44433957 Ki = 112 nM T99041 CI15HN 44433958 Ki = 152 nM T99041 C1C9SZ 44433959 Ki = 1944 nM T99041 CA4VY1 44433960 Ki = 3311 nM T99041 CU69GM 44433961 Ki > 10000 nM T99041 CDF80C 44433962 Ki > 10000 nM T99041 CKN0C1 44433969 Ki = 3081 nM T99041 C53UEG 44434115 IC50 = 8 nM T99041 CE92DA 44435310 IC50 = 261000 nM T99041 C3SBK5 44435313 IC50 = 8000 nM T99041 CX7UN0 44435314 IC50 = 4200 nM T99041 CE7XI5 44435315 IC50 > 50000 nM T99041 CGAR49 44435316 IC50 > 250000 nM T99041 C17HRW 44439324 IC50 = 127 nM T99041 C1JQ8Y 44439325 IC50 = 47.6 nM T99041 CAOY46 44439326 IC50 = 13.9 nM T99041 C8XU3A 44439327 IC50 = 57.5 nM T99041 CI7SP9 44439328 IC50 = 10.9 nM T99041 CWG07L 44439329 IC50 = 30.5 nM T99041 CT9V8F 44439330 IC50 = 21 nM T99041 C74ANZ 44439331 IC50 = 13.5 nM T99041 C4B5DI 44439332 IC50 = 12.2 nM T99041 C7LEY1 44439333 IC50 = 8.7 nM T99041 CCJ8T1 44439334 IC50 = 4.1 nM T99041 CWU62R 44439335 IC50 = 10.8 nM T99041 CWG89M 44439336 IC50 = 8.2 nM T99041 CEL4H9 44439337 IC50 = 1.6 nM T99041 C4H3EF 44439338 IC50 = 4.3 nM T99041 C3MLU4 44439339 IC50 = 6.8 nM T99041 C8P1AX 44439340 IC50 = 3 nM T99041 C54TPV 44439341 IC50 = 1.3 nM T99041 CEP51V 44439342 IC50 = 5.6 nM T99041 C4YWH2 44439343 IC50 = 2.3 nM T99041 C1G5PI 44439344 IC50 = 2.4 nM T99041 C02LBF 44439345 IC50 = 2.7 nM T99041 CBE1D5 44439346 IC50 = 3.1 nM T99041 C5T7XF 44439347 IC50 = 2.5 nM T99041 CMC8H4 44439348 IC50 = 1.6 nM T99041 CX4MT0 44439350 IC50 = 1.5 nM T99041 C0OJ1T 44439353 IC50 = 1 nM T99041 C9T6FK 44439354 IC50 = 1.2 nM T99041 C69XIH 44439668 IC50 = 990 nM T99041 CDF76U 44439670 IC50 = 500 nM T99041 C6E8JI 44440627 Ki = 2700 nM T99041 CUQ7K0 44440629 Ki = 280 nM T99041 CSXH19 44440630 Ki = 610 nM T99041 CSI93Z 44440631 Ki = 490 nM T99041 COP6M3 44440633 Ki = 790 nM T99041 C5GKC8 44440634 Ki = 210 nM T99041 CTI8C4 44440635 Ki = 430 nM T99041 C2VAG9 44440645 Ki = 17 nM T99041 CTQR78 44440647 Ki = 20 nM T99041 C08ZST 44440659 Ki = 1 nM T99041 CA9WC3 44440660 Ki = 85 nM T99041 CXC50E 44440661 Ki = 7 nM T99041 CR3PM7 44440662 Ki = 1.7 nM T99041 CB4Q0H 44440663 Ki = 3.4 nM T99041 C6YEQ8 44440664 Ki = 9 nM T99041 CCSI57 44440665 Ki = 1.3 nM T99041 CR4B1M 44443293 IC50 = 30 nM T99041 CY16JP 44443294 IC50 = 38 nM T99041 CN24IJ 44443296 IC50 = 40 nM T99041 C8DSC1 44443297 IC50 = 42 nM T99041 C4F5JW 44443298 IC50 = 47 nM T99041 CJ0G3N 44443299 IC50 = 49 nM T99041 C9F7NQ 44443300 IC50 = 62 nM T99041 C7QCO2 44443301 IC50 = 79 nM T99041 CCQ82F 44443302 IC50 = 86 nM T99041 C1M5TF 44443309 IC50 = 27 nM T99041 CSAE59 44443313 IC50 = 50 nM T99041 CK5E8V 44443319 IC50 = 69 nM T99041 CD0NM4 44443335 IC50 = 78 nM T99041 CEF6H5 44443336 IC50 = 80 nM T99041 CTIM25 44443338 IC50 = 81 nM T99041 CE9Q7A 44443341 IC50 = 83 nM T99041 CI8Q5O 44443343 IC50 = 91 nM T99041 C0MOV3 44443346 IC50 = 2.4 nM T99041 C52VPZ 44443347 IC50 = 3.2 nM T99041 CJ8P7U 44443348 IC50 = 3.3 nM T99041 C8U1XN 44443349 IC50 = 3.6 nM T99041 CM5WU9 44443350 IC50 = 5.3 nM T99041 CB9IM0 44443351 IC50 = 5.4 nM T99041 C8WI4F 44443352 IC50 = 6.2 nM T99041 C3NI8P 44443353 IC50 = 6.7 nM T99041 C7M0HV 44443354 IC50 = 8.5 nM T99041 C0UG4R 44443355 IC50 = 10 nM T99041 C7B5HK 44443356 IC50 = 10 nM T99041 C2G1PX 44443357 IC50 = 3 nM T99041 C3AUF2 44443358 IC50 = 3.4 nM T99041 C0WO5B 44443359 IC50 = 3.5 nM T99041 CUG6X5 44443360 IC50 = 5.5 nM T99041 CARK80 44443361 IC50 = 5.3 nM T99041 CP7WL5 44443363 IC50 = 1.1 nM T99041 C4V0SN 44443364 IC50 = 4.7 nM T99041 CQL53Y 44443365 IC50 = 46 nM T99041 CD2L9G 44443366 IC50 = 3.8 nM T99041 CPN7J9 44443420 IC50 = 65 nM T99041 CI4VR8 44443421 IC50 > 3 nM T99041 CA0NZ7 44443707 IC50 = 140 nM T99041 C24ZHB 44443708 IC50 = 150 nM T99041 C8R4OD 44443709 IC50 = 130 nM T99041 CLDN63 44443710 IC50 = 180 nM T99041 C7LNP2 44443711 IC50 = 230 nM T99041 CJX2M7 44443712 IC50 = 220 nM T99041 C6RST0 44443713 IC50 = 260 nM T99041 C3YL9X 44443714 IC50 = 250 nM T99041 CRH8M1 44443715 IC50 = 250 nM T99041 CIB50E 44443717 IC50 = 130 nM T99041 CK6QF4 44443719 IC50 = 280 nM T99041 CX6O1P 44443720 IC50 = 65 nM T99041 C0YV2D 44443723 IC50 = 610 nM T99041 C1BUJ5 44443725 IC50 = 570 nM T99041 CXS34I 44443727 IC50 = 50 nM T99041 CCHS17 44443729 IC50 = 110 nM T99041 C39KZG 44443736 IC50 = 250 nM T99041 C5H8EJ 44443737 IC50 = 370 nM T99041 CS3Y1G 44444344 IC50 = 100 nM T99041 CL2U9C 44444352 IC50 = 68 nM T99041 C8VE5T 44444353 IC50 = 274 nM T99041 C8F5HC 44444371 IC50 = 4 nM T99041 CEW50M 44444373 IC50 = 4 nM T99041 CO0M7Y 44444375 IC50 = 7 nM T99041 CS93BI 44444377 IC50 = 12 nM T99041 C9J4FB 44444379 IC50 = 14 nM T99041 C3YA4K 44444383 IC50 = 18 nM T99041 C75OIP 44444386 IC50 = 2 nM T99041 C4J6ZG 44444390 IC50 = 4 nM T99041 C05EBU 44444391 IC50 = 2 nM T99041 CSN27E 44445042 IC50 = 5.7 nM T99041 CGN61Q 44445047 IC50 = 1.5 nM T99041 CYW8E3 44445051 IC50 = 2.8 nM T99041 CRG64M 44445053 IC50 = 0.66 nM T99041 C6ZID3 44445055 IC50 = 0.43 nM T99041 C72KOR 44445057 IC50 = 438 nM T99041 C0RTA6 44445060 IC50 = 0.46 nM T99041 CIK8G3 44445063 IC50 = 0.32 nM T99041 CN05VX 44445065 IC50 = 6.3 nM T99041 COA90R 44445067 IC50 = 132 nM T99041 CHRX61 44445075 IC50 > 36900 nM T99041 C6C5IN 44448853 IC50 = 559 nM T99041 CB7MS5 44448857 IC50 = 582 nM T99041 C4IXY7 44448987 IC50 = 2 nM T99041 COP51N 44448988 IC50 = 1 nM T99041 C8KW2A 44448989 IC50 = 99 nM T99041 C9ZRP1 44449015 IC50 = 19 nM T99041 C7E4ZI 44449016 IC50 = 107 nM T99041 CKM5H1 44449017 IC50 = 52 nM T99041 CJ2WY0 44449038 IC50 = 4 nM T99041 C8F2SQ 44449064 IC50 = 2 nM T99041 C7PBF3 44449092 IC50 = 15 nM T99041 CUM32L 44449149 IC50 = 1 nM T99041 CK5M4R 44451509 IC50 = 56 nM T99041 CWI3J9 44451511 IC50 = 41 nM T99041 CEFD93 44451512 IC50 = 600 nM T99041 CKCF72 44451863 IC50 = 51 nM T99041 CR51UD 44451910 IC50 = 60 nM T99041 C76NDG 44451911 IC50 = 16 nM T99041 C20LHD 44452002 IC50 = 13000 nM T99041 CODZ87 44452030 IC50 = 110 nM T99041 CV0Z4T 44452035 IC50 = 70 nM T99041 C7RI2V 44452075 IC50 = 16 nM T99041 CUC93Q 44452076 IC50 = 1100 nM T99041 CK5DW6 44453458 IC50 = 30 nM T99041 C3X8BJ 44453460 IC50 = 42 nM T99041 CDF8R2 44453520 IC50 = 50000 nM T99041 CVO9F2 44453648 IC50 = 57 nM T99041 C91FSI 44453672 IC50 = 90 nM T99041 C5UET4 44453690 IC50 = 645 nM T99041 C2JE8C 44453692 IC50 = 1165 nM T99041 C6EC4J 44453922 IC50 = 12 nM T99041 C4C6NK 44453968 IC50 = 93 nM T99041 CDS52W 44453970 IC50 = 3.2 nM T99041 C9V2HU 44454016 IC50 = 50 nM T99041 CW4H0F 44455959 IC50 = 52 nM T99041 C0S2TV 44455961 IC50 = 21 nM T99041 CH04ND 44455993 IC50 = 37 nM T99041 C50MTS 44456000 IC50 = 604 nM T99041 CQF6O5 44456002 IC50 = 620 nM T99041 CFZB21 44456030 IC50 = 1900 nM T99041 CI0K1D 44456032 IC50 = 340 nM T99041 CYN5Z3 44456147 IC50 = 310 nM T99041 C1WBL5 44456148 IC50 = 350 nM T99041 C3HE5Z 44456310 IC50 = 670 nM T99041 CHKT64 44458509 IC50 = 830 nM T99041 CXWQ16 44458510 IC50 = 360 nM T99041 CBSZ02 44458521 IC50 = 88 nM T99041 CIA6J1 44458523 IC50 = 56 nM T99041 C6LKZ7 44458534 IC50 = 27 nM T99041 CR41OX 44458540 IC50 = 870 nM T99041 CNK09O 44458542 IC50 = 70 nM T99041 CM65HC 44458548 IC50 = 23 nM T99041 CKM0F5 44458549 IC50 = 75 nM T99041 CR4CP3 44458554 IC50 = 21 nM T99041 CU68KW 44458566 IC50 = 270 nM T99041 CC7I6Y 44458573 IC50 = 110 nM T99041 CCI52U 44458574 IC50 = 250 nM T99041 C0K7EZ 44458575 IC50 = 210 nM T99041 CNK64C 44458581 IC50 = 250 nM T99041 CF7I9V 44458586 IC50 = 67 nM T99041 CW7QX0 44458587 IC50 = 55 nM T99041 CJ7Y6A 44458592 IC50 = 35 nM T99041 C9QMB2 44458594 Ki = 56 nM T99041 CPJW14 44458603 Ki = 128 nM T99041 C0K2SV 44458617 Ki = 28 nM T99041 CSIL15 44458629 IC50 = 54 nM T99041 C3EZ1V 44458770 IC50 = 89 nM T99041 COHJ95 44560137 IC50 = 252 nM T99041 CAY0V7 44560138 IC50 = 7.3 nM T99041 C8LNP1 44560139 IC50 = 6.2 nM T99041 CUJR76 44560140 IC50 = 22 nM T99041 C0V4UW 44560141 IC50 = 8.6 nM T99041 CFX7Y2 44560154 IC50 = 12 nM T99041 CGW57E 44560155 IC50 = 88 nM T99041 C0Z5AB 44560156 IC50 = 16 nM T99041 C9JL5Y 44560157 IC50 = 27 nM T99041 C4NC6K 44560158 IC50 = 2.9 nM T99041 CHJ2I3 44560159 IC50 = 7.8 nM T99041 CR4AD0 44560160 IC50 = 8.7 nM T99041 CO9I7S 44560169 IC50 = 13 nM T99041 CD6H2S 44560170 IC50 > 316 nM T99041 C9QC1W 44560171 IC50 = 33 nM T99041 CNF05Y 44560172 IC50 = 3.1 nM T99041 CB73HS 44560173 IC50 = 2.6 nM T99041 CC9B5Y 44560174 IC50 = 3.3 nM T99041 C41LTG 44560184 IC50 = 4.1 nM T99041 C7E1TG 44560185 IC50 = 3.1 nM T99041 C8Z2AR 44560186 IC50 = 3.1 nM T99041 CX3EK8 44560187 IC50 = 8.3 nM T99041 C1BX6I 44560188 IC50 = 5.3 nM T99041 CY78ZH 44560250 IC50 = 2.8 nM T99041 CR69YS 44560251 IC50 = 2.7 nM T99041 C60VSL 44560252 IC50 = 2.4 nM T99041 C70CYA 44560253 IC50 = 8.2 nM T99041 C8CED7 44560254 IC50 = 4.5 nM T99041 CC09EL 44560255 IC50 = 5.4 nM T99041 C5MN2V 44560265 IC50 = 2.9 nM T99041 C75KOL 44560266 IC50 = 5.7 nM T99041 CED9I6 44560267 IC50 = 5.8 nM T99041 C9DLI3 44560268 IC50 = 13 nM T99041 CU65ER 44560279 IC50 = 109 nM T99041 C17LFS 44560280 IC50 = 75 nM T99041 CTD6U0 44560281 IC50 = 31 nM T99041 CB7V0P 44560282 IC50 > 316 nM T99041 CJ4EN1 44560283 IC50 = 39 nM T99041 C91DWY 44560396 IC50 > 100000 nM T99041 CZ9WJ0 44560397 IC50 > 100000 nM T99041 C0FLU7 44560398 IC50 = 80100 nM T99041 CZ43JR 44560454 IC50 > 100000 nM T99041 CY38QP 44560549 IC50 > 100000 nM T99041 C7IL3K 44560550 IC50 > 100000 nM T99041 CF9J7Z 44560551 IC50 > 100000 nM T99041 C1QAI4 44560552 IC50 > 100000 nM T99041 CK25CG 44560553 IC50 > 50000 nM T99041 C4C9NG 44560554 IC50 > 100000 nM T99041 CKIH45 44560555 IC50 > 100000 nM T99041 C2LW3C 44560595 IC50 > 100000 nM T99041 C47WCK 44560596 IC50 > 100000 nM T99041 CL8AE5 44560597 IC50 > 100000 nM T99041 C1YJ8C 44560648 IC50 > 50000 nM T99041 CY6GU1 44560649 IC50 > 62500 nM T99041 C12EYZ 44560650 IC50 = 178000 nM T99041 C7LY9V 44560651 IC50 > 31250 nM T99041 CG5CB2 44560698 IC50 > 250000 nM T99041 CR56BA 44560699 IC50 = 4970 nM T99041 CAK3U5 44560701 IC50 > 100000 nM T99041 C5OW2C 44560747 IC50 > 500000 nM T99041 CM2GN5 44560748 IC50 > 1000000 nM T99041 C5FSB4 44560749 IC50 > 500000 nM T99041 C5WEG1 44560750 IC50 > 250000 nM T99041 CN0KO4 44560770 IC50 = 22 nM T99041 CZSO82 44560823 Ki = 4900 nM T99041 C4IVD9 44560824 IC50 = 37000 nM T99041 C4L3VZ 44560825 IC50 = 15600 nM T99041 CHV7S1 44560826 IC50 = 9700 nM T99041 CE3NF4 44560849 IC50 = 12700 nM T99041 CT6P5E 44560850 IC50 = 16800 nM T99041 CTH9P2 44560851 Ki = 1200 nM T99041 CGZ48C 44560928 IC50 = 51000 nM T99041 C9EK8A 44560929 IC50 > 1000000 nM T99041 CM68VD 44560930 IC50 = 3700 nM T99041 C4SMJ1 44560961 IC50 = 35 nM T99041 C2I3TR 44560962 IC50 = 340 nM T99041 CGV49L 44560963 IC50 = 290 nM T99041 CY0L1G 44560964 IC50 = 2200 nM T99041 C7FST1 44560988 IC50 = 530 nM T99041 CGOM86 44560989 IC50 = 52000 nM T99041 C74ZNK 44560990 IC50 = 2500 nM T99041 C95AUS 44560991 IC50 = 560 nM T99041 CTJ23N 44561008 IC50 = 1300 nM T99041 CR2A0E 44561009 IC50 = 253 nM T99041 C4LQY2 44561010 IC50 = 107 nM T99041 C28XDF 44561011 IC50 = 71 nM T99041 CQ04BE 44561046 IC50 = 9800 nM T99041 C8IF7B 44561117 IC50 = 9200 nM T99041 C29VDX 44561118 IC50 = 200 nM T99041 CB4JA7 44561119 IC50 = 8800 nM T99041 C5K9CX 44561120 IC50 = 55 nM T99041 CQ8DN4 44561152 IC50 = 4400 nM T99041 C4DBU1 44561153 IC50 = 615 nM T99041 C73WBR 44561154 IC50 = 600 nM T99041 CJ91UC 44561155 IC50 = 46 nM T99041 CMO6S2 44561191 IC50 = 20 nM T99041 CF9SB3 44561192 IC50 = 40 nM T99041 C5X1VJ 44561193 IC50 = 120 nM T99041 C31GMV 44561194 IC50 = 85 nM T99041 C1U4YQ 44565237 IC50 = 27 nM T99041 CRK69O 44565238 IC50 = 19 nM T99041 C6M2WD 44565239 IC50 = 21 nM T99041 CTZ9L0 44565254 IC50 = 22 nM T99041 CEMV93 44565274 IC50 = 26 nM T99041 C5E6PQ 44565275 IC50 = 17 nM T99041 CI93OK 44565276 IC50 = 20 nM T99041 C2HRF1 44565277 IC50 = 26 nM T99041 CFEC28 44565466 IC50 = 85 nM T99041 C5MON6 44565467 IC50 = 54 nM T99041 CGA4U6 44565488 IC50 = 64 nM T99041 C1BZ3I 44565489 IC50 = 84 nM T99041 CP3C5F 44565490 IC50 = 75 nM T99041 CRU86T 44565491 IC50 = 62 nM T99041 C3C2DL 44565492 IC50 = 85 nM T99041 CJ2W1P 44565512 IC50 = 60 nM T99041 C5Z9GW 44565513 IC50 = 73 nM T99041 C3I0MO 44565514 IC50 = 86 nM T99041 CI3J6Y 44565535 IC50 = 68 nM T99041 CB90XZ 44565536 IC50 = 101 nM T99041 C01SLH 44565537 IC50 = 24 nM T99041 C8Y2LX 44565538 IC50 = 10 nM T99041 CXD19F 44565539 IC50 = 56 nM T99041 C5BIY6 44565582 IC50 = 309 nM T99041 CFK92H 44565583 IC50 = 25 nM T99041 CE3UT4 44565584 IC50 = 309 nM T99041 CA0O7F 44565585 IC50 = 41 nM T99041 C7LPW8 44565586 IC50 = 134 nM T99041 C39RGP 44565611 IC50 = 338 nM T99041 CPZ7J3 44565844 IC50 = 8.7 nM T99041 C9BGR3 44565845 IC50 = 8.2 nM T99041 CR83QA 44565869 IC50 = 7.4 nM T99041 C6K2WL 44565870 IC50 = 5.6 nM T99041 C3UL2E 44565871 IC50 = 5.2 nM T99041 C9SL5D 44565872 IC50 = 4.8 nM T99041 CZBX95 44565889 IC50 = 31 nM T99041 C1TLY0 44565890 IC50 = 51 nM T99041 CEO20N 44565891 IC50 = 31 nM T99041 COA7X5 44565892 IC50 = 13 nM T99041 CRO3D2 44567651 IC50 = 186 nM T99041 CM95OD 44567652 IC50 = 221 nM T99041 CX6WL5 44567653 IC50 = 27 nM T99041 C4MP9D 44567654 IC50 = 49 nM T99041 CV23FP 44567668 IC50 = 85 nM T99041 CD4C7Y 44567710 IC50 = 123 nM T99041 C4CUJ6 44567711 IC50 = 147 nM T99041 CK1C7W 44567712 IC50 = 78 nM T99041 CTK1I9 44567713 IC50 = 91 nM T99041 C9LQ7N 44567714 IC50 = 1300 nM T99041 CM50CU 44567747 IC50 = 93 nM T99041 C9IF5L 44567748 IC50 > 10000 nM T99041 CMGJ56 44567749 Ki = 5 nM T99041 CR43EI 44567750 Ki = 12 nM T99041 CZ3G4I 44567783 Ki = 31 nM T99041 CNA0I9 44567918 IC50 = 165 nM T99041 C6BXT0 44567919 IC50 = 153 nM T99041 CJ85MG 44567920 IC50 = 110 nM T99041 CUJD19 44567976 IC50 = 38 nM T99041 C5YB6E 44567977 IC50 = 95 nM T99041 CNF09E 44567978 IC50 = 152 nM T99041 C70WEI 44567979 IC50 = 59 nM T99041 CJ0YL5 44568015 IC50 = 2540 nM T99041 CW7NB6 44568016 IC50 = 109 nM T99041 CY8Z3F 44568017 IC50 = 229 nM T99041 CRM76D 44568018 IC50 = 95 nM T99041 C7D4EP 44568055 IC50 = 3430 nM T99041 C3E2UC 44568056 IC50 = 3740 nM T99041 CCG83U 44568057 IC50 = 51 nM T99041 C8XW9A 44568058 IC50 = 31 nM T99041 CMQ7D5 44568097 IC50 = 42 nM T99041 C1F9OL 44568098 IC50 = 63 nM T99041 CUYK75 44568099 IC50 = 92 nM T99041 CZ81XF 44568100 IC50 = 141 nM T99041 C6GT0A 44568134 IC50 = 422 nM T99041 C6IW5D 44568135 IC50 = 630 nM T99041 C3PWD8 44568136 IC50 = 118 nM T99041 C3JBY7 44568137 IC50 = 1715 nM T99041 C4NCA7 44568169 IC50 = 84 nM T99041 C8TXH9 44568170 IC50 = 181 nM T99041 C17PZX 44568171 IC50 = 146 nM T99041 C7SCJ1 44568172 IC50 = 186 nM T99041 CT10GB 44571684 IC50 = 1440 nM T99041 CAT7M0 44571686 IC50 = 510 nM T99041 CSU97M 44571688 IC50 = 3400 nM T99041 C8UGS0 44571690 IC50 = 490 nM T99041 C2WC7S 44571735 IC50 = 410 nM T99041 C0BX2S 44571737 IC50 = 490 nM T99041 C7KYX8 44571739 IC50 = 1392 nM T99041 C2ZYC9 44571741 IC50 = 1500 nM T99041 C68DZI 44571781 IC50 = 350 nM T99041 C1HSU7 44571783 IC50 = 3100 nM T99041 C5WDE4 44571785 IC50 = 405 nM T99041 CB20PW 44571787 IC50 = 387 nM T99041 C8NB2X 44571851 IC50 = 6400 nM T99041 C40YLT 44571853 IC50 = 597 nM T99041 CV9BW0 44571855 IC50 = 423 nM T99041 C0LMD8 44571898 IC50 = 239 nM T99041 CLFG01 44571900 IC50 = 788 nM T99041 C1U5MS 44571902 IC50 = 180 nM T99041 C8DAK4 44571945 IC50 = 288 nM T99041 CM9DP7 44571947 IC50 = 150 nM T99041 CZCU54 44571949 IC50 = 50 nM T99041 CJ96CO 44571951 IC50 = 67 nM T99041 CQW5N2 44571996 IC50 = 260 nM T99041 C7E6IB 44572718 IC50 = 298 nM T99041 CUH81Y 44572719 IC50 = 2 nM T99041 CJHR19 44572720 IC50 = 10 nM T99041 CG71OU 44572782 IC50 = 1600 nM T99041 CG86WR 44580460 IC50 = 13000 nM T99041 C7NP1S 44580497 IC50 = 12000 nM T99041 CQU6S5 44580498 IC50 = 50000 nM T99041 C9JY0C 44580499 IC50 = 180000 nM T99041 CT1N3H 44580500 IC50 = 390000 nM T99041 CYO50L 44580540 IC50 = 11 nM T99041 CSX3I9 44580589 IC50 = 25 nM T99041 CGB0H3 44580664 IC50 = 21 nM T99041 CPR2S7 44589876 IC50 = 7800 nM T99041 C3H0AD 44589877 IC50 = 1000 nM T99041 CY5TC1 44589878 IC50 = 2200 nM T99041 CKM0Z1 44589879 IC50 = 870 nM T99041 CPU4J0 44589931 IC50 = 2500 nM T99041 C4X9GH 44589932 IC50 = 3300 nM T99041 C2DQ0C 44589933 IC50 = 570 nM T99041 C27TUB 44589934 IC50 = 470 nM T99041 CUZ3P0 44589935 IC50 = 190 nM T99041 CM18AD 44589985 IC50 = 64 nM T99041 C4LEZ6 44589986 IC50 = 13 nM T99041 CW2T9J 44589987 IC50 = 12 nM T99041 C1SK7V 44590037 IC50 = 2.7 nM T99041 C6NE1Y 44590038 IC50 = 3.3 nM T99041 CGV2A7 44590039 IC50 = 270 nM T99041 C1KC3N 44590040 IC50 = 35 nM T99041 CZGQ12 44590126 IC50 = 130 nM T99041 CV7RD4 44590127 IC50 = 70 nM T99041 CIE7S0 44590128 IC50 = 350 nM T99041 CCK2S8 44590129 IC50 = 1 nM T99041 C39MKI 44590183 IC50 = 0.64 nM T99041 C82PIC 44590184 IC50 = 1.9 nM T99041 C85SFW 44590185 IC50 = 0.79 nM T99041 C48MPJ 44590596 IC50 = 251 nM T99041 CYE25R 44590598 Ki = 3.6 nM T99041 CI98LA 44590648 IC50 = 22 nM T99041 CBAH06 44590649 IC50 = 6.2 nM T99041 C5R9NI 44590650 IC50 = 0.13 nM T99041 C0W2FC 44590651 IC50 = 0.15 nM T99041 CRN4U5 44590696 IC50 = 4.3 nM T99041 CTC24F 44590734 IC50 = 8 nM T99041 C8CRO4 44590736 IC50 = 18 nM T99041 C91FTW 44591848 IC50 = 18 nM T99041 CY78PR 44591849 IC50 = 22 nM T99041 CE2LW5 44591850 IC50 = 27 nM T99041 CZW0V4 44592369 IC50 > 30000 nM T99041 C3WJ6O 44592370 IC50 = 1930 nM T99041 C07LHO 44592439 IC50 = 3580 nM T99041 CTC4G9 44592440 IC50 > 30000 nM T99041 CIVD36 44592441 IC50 = 25900 nM T99041 C65OXJ 44592442 IC50 > 30000 nM T99041 C8Z0CX 44592443 IC50 = 3250 nM T99041 C9PL5R 44592444 IC50 = 1420 nM T99041 C7L8UN 44592445 IC50 > 30000 nM T99041 CQG62W 44592506 IC50 = 1970 nM T99041 CQHL54 44592507 IC50 = 272 nM T99041 CV42SK 44592508 IC50 = 270 nM T99041 C82YQS 44592509 IC50 = 35 nM T99041 CWJ2U0 44592510 IC50 = 26 nM T99041 CQI40A 44592511 IC50 = 19 nM T99041 CY8R3Q 44593399 IC50 = 115000 nM T99041 CP8YC3 44593408 IC50 = 161000 nM T99041 C4L6NS 44593409 IC50 = 245000 nM T99041 CI0FT1 44593463 IC50 = 47 nM T99041 CAWO01 44593726 IC50 = 6030 nM T99041 CY7Q8W 44629524 IC50 = 22 nM T99041 C65KPR 45101722 IC50 = 6.3 nM T99041 CXYT36 45101723 IC50 = 3 nM T99041 C2RNP7 45102670 IC50 = 16 nM T99041 CQ85WF 45263621 Ki = 6 nM T99041 CGZD98 45265711 IC50 = 103 nM T99041 CW09DZ 45265891 Ki = 3.2 nM T99041 CCO76A 45266134 IC50 = 1700 nM T99041 CU4C5P 45266135 IC50 = 20 nM T99041 CLVM20 45266136 IC50 = 19 nM T99041 CIS3Z8 45267371 IC50 = 92 nM T99041 C8H9GV 45267527 IC50 = 3.2 nM T99041 CP9B0W 45267530 IC50 = 15 nM T99041 C3GJK0 45267531 IC50 = 5.4 nM T99041 CD67HE 45268222 IC50 = 47 nM T99041 CN38QU 45268229 IC50 = 12 nM T99041 CEQ16V 45268233 IC50 = 8 nM T99041 CT93EB 45268323 IC50 = 27 nM T99041 C0QB1V 45268417 IC50 = 2 nM T99041 C2S9ZT 45268436 IC50 = 27 nM T99041 C60MVX 45269112 IC50 = 66 nM T99041 CV7IL1 45269122 IC50 = 24 nM T99041 CX8WC0 45269123 IC50 = 30 nM T99041 C9HR0K 45269274 IC50 = 7.8 nM T99041 CZ1N2O 45269275 IC50 = 12 nM T99041 CIE21V 45269276 IC50 = 5.6 nM T99041 C2W6MT 45269961 IC50 = 87 nM T99041 CWT60M 45269971 IC50 = 14 nM T99041 C4CG2K 45269976 IC50 = 27 nM T99041 CK5P9W 45269994 IC50 = 152 nM T99041 C2A8WO 45269995 IC50 > 16000 nM T99041 C8QJ7X 45270108 IC50 = 7.1 nM T99041 CYWK62 45270115 IC50 = 10 nM T99041 C6E7PR 45270793 IC50 = 92 nM T99041 C6B0CO 45270800 IC50 = 20 nM T99041 CS89DP 45270806 IC50 = 53 nM T99041 CZI9A4 45270821 IC50 > 1600 nM T99041 CQM4X3 45270889 IC50 = 49 nM T99041 CGF7Z6 45270958 IC50 = 2.7 nM T99041 CH5S8Y 45270959 IC50 = 2.2 nM T99041 CM80NZ 45271662 IC50 > 1600 nM T99041 C5NH6Q 45271791 IC50 = 4 nM T99041 C8Z3DK 45271794 IC50 = 3.9 nM T99041 CX62YA 45271796 IC50 = 1.3 nM T99041 CZ8EO2 45271803 IC50 = 3.5 nM T99041 CJ7Q9E 45271813 IC50 = 6.8 nM T99041 CLSJ45 45272523 IC50 = 77 nM T99041 C75XKZ 45272524 IC50 = 27 nM T99041 CSC67Y 45272544 IC50 > 16000 nM T99041 CJI2R6 45272664 IC50 = 2.3 nM T99041 C49BKQ 45272672 IC50 = 5.9 nM T99041 CP36CT 45272682 IC50 = 1.5 nM T99041 C8NL4U 45272683 IC50 = 2.7 nM T99041 CI5AU6 45273390 IC50 = 94 nM T99041 C6S0OC 45273404 IC50 = 8 nM T99041 C2EK3O 45273409 IC50 = 53 nM T99041 C1ZX6U 45273413 IC50 > 1600 nM T99041 CYMR87 45273573 IC50 = 3.5 nM T99041 CFL87A 45273581 IC50 = 6.3 nM T99041 C2XB0P 45273589 IC50 = 6.1 nM T99041 C28PRV 45273594 IC50 = 4.8 nM T99041 CSX2T9 45273602 IC50 = 3.7 nM T99041 CMP59Q 45273603 IC50 = 1.1 nM T99041 C2R3QM 45481268 IC50 = 9 nM T99041 C31XRV 45482320 IC50 = 14130 nM T99041 C28ZXW 45487888 IC50 = 2 nM T99041 C74SVC 45487893 IC50 = 31 nM T99041 C2N3IZ 45487894 IC50 = 3 nM T99041 CP62TC 45487898 IC50 = 4 nM T99041 CPBA81 45487901 IC50 = 90 nM T99041 C0SQW3 45487902 IC50 = 62 nM T99041 CWQ1R9 45487903 IC50 = 2 nM T99041 C8H1KY 45487904 IC50 = 4 nM T99041 C1LJR6 45487907 IC50 = 120 nM T99041 C6X7WJ 45487908 IC50 = 4 nM T99041 CZDS09 45487910 IC50 = 76 nM T99041 CNVU49 45487911 IC50 = 180 nM T99041 C5OXM9 45487915 IC50 = 17 nM T99041 CPJ19X 45487917 IC50 = 2 nM T99041 C16DIR 45487918 IC50 = 28 nM T99041 CV2R7M 45487920 IC50 = 1 nM T99041 C57JRG 45487921 IC50 = 11 nM T99041 C4JD1P 45487922 IC50 = 32 nM T99041 CH30BL 45487925 IC50 = 130 nM T99041 CPB85R 45487926 IC50 = 17 nM T99041 CTY16E 45487930 IC50 = 7 nM T99041 C4QTL9 45487931 IC50 = 5 nM T99041 CG9V0L 45487940 IC50 = 22 nM T99041 C5XTV1 45487945 IC50 = 10 nM T99041 C3VK4G 45487946 IC50 = 2 nM T99041 C0SNL2 46209134 IC50 = 1.6 nM T99041 CE9M5C 46209244 IC50 = 1.6 nM T99041 CW60IG 46209246 IC50 = 1.6 nM T99041 CV65TL 46216691 IC50 = 11 nM T99041 C4QO6X 46216692 IC50 = 0.5 nM T99041 C4GPM1 46229765 IC50 = 61 nM T99041 CCO56J 46229809 IC50 = 38 nM T99041 C0CQM4 46229810 IC50 = 5500 nM T99041 CQ5S8A 46229811 IC50 = 0.5 nM T99041 C6K1YR 46229812 IC50 = 1.7 nM T99041 CU4GE7 46230652 IC50 = 53000 nM T99041 CI4A3C 46230653 IC50 = 19 nM T99041 CEPY06 46231493 IC50 = 1.2 nM T99041 CIEK51 46842529 IC50 = 2810 nM T99041 CDP7Q4 46870369 IC50 = 17 nM T99041 CPH7B4 46871723 IC50 = 8 nM T99041 CDBC45 46890720 IC50 = 180 nM T99041 CLK47C 46890721 IC50 = 23 nM T99041 CS6HL3 46890722 IC50 = 50 nM T99041 C2JY6P 46890723 IC50 = 24 nM T99041 CP7C1L 46890780 IC50 = 26 nM T99041 CED80Z 46890852 IC50 = 93 nM T99041 CA3PE4 46890853 IC50 = 160 nM T99041 CY9T8W 46890854 IC50 = 66 nM T99041 C3TJ0H 46890912 IC50 = 27 nM T99041 CT9HQ6 46890913 IC50 = 24 nM T99041 C9IP7B 46890914 IC50 = 18 nM T99041 CSZE87 46891193 IC50 = 12 nM T99041 C18UES 46891235 IC50 = 59 nM T99041 C23LCY 46891237 IC50 = 65 nM T99041 C57UXS 46891239 IC50 = 80 nM T99041 CIM3K6 46891241 IC50 = 204 nM T99041 C4AUV2 46891291 IC50 = 326 nM T99041 C0UKG7 46891293 IC50 = 121 nM T99041 CJ4G6X 46891342 IC50 = 32 nM T99041 CAL9K6 46891534 IC50 = 15 nM T99041 CPN5T2 46891535 IC50 = 71 nM T99041 C4XTW7 46893990 IC50 > 100000 nM T99041 C8O5VR 46899592 Ki = 8.7 nM T99041 CTY0M5 46899593 Ki = 1 nM T99041 CK9TH1 46899594 Ki = 3.1 nM T99041 C8XD0Q 46899595 Ki = 0.2 nM T99041 CZ84ST 46899596 Ki = 0.5 nM T99041 CPZ70E 46899597 Ki = 0.3 nM T99041 CD3IJ8 46899752 Ki = 0.9 nM T99041 CRK59N 46899753 Ki = 6.6 nM T99041 C6LXU5 46899754 Ki = 2 nM T99041 C52JZL 46899755 Ki = 0.6 nM T99041 C4RC1S 46899756 Ki = 1.8 nM T99041 CP84HR 46899757 Ki = 3.8 nM T99041 CBV4W0 46899937 Ki = 2.6 nM T99041 C5QEJ4 46899938 Ki = 1.1 nM T99041 CHR6V9 46899939 Ki = 2 nM T99041 CQ3A8F 46899940 Ki = 3.2 nM T99041 CX2P8Z 46899941 Ki = 0.7 nM T99041 CC2X1J 46899942 Ki = 2.6 nM T99041 C5QA9M 46900103 Ki = 4 nM T99041 CBI0Q2 46900104 Ki = 0.9 nM T99041 C4IU2E 46900105 Ki = 5 nM T99041 CZEB71 46900106 Ki = 4.7 nM T99041 C2TJW5 46900108 Ki = 1.5 nM T99041 C54ATK 46900259 Ki = 1.3 nM T99041 CI3P6J 46900261 Ki = 2.4 nM T99041 C6DP2G 46900418 Ki = 3.1 nM T99041 CP50DR 46900420 Ki = 5 nM T99041 CF3BL8 46905362 IC50 = 1500 nM T99041 C9JKO5 46905992 IC50 = 21 nM T99041 C8DSG7 46916343 IC50 > 100000 nM T99041 C3RO8F 46916345 IC50 > 100000 nM T99041 CX07LJ 46916346 IC50 > 100000 nM T99041 CF94MW 46916347 IC50 > 100000 nM T99041 CH3F7O 46916384 IC50 > 100000 nM T99041 CM8W6E 46916385 IC50 > 100000 nM T99041 C6FA9Q 46916386 IC50 > 100000 nM T99041 CAW86J 46916387 IC50 > 100000 nM T99041 C63HBE 46916388 IC50 > 100000 nM T99041 CD1CZ7 46916389 IC50 > 100000 nM T99041 CH80LK 46916433 IC50 > 100000 nM T99041 CN4A3P 46916435 IC50 > 100000 nM T99041 CUQ86M 46917047 IC50 > 100000 nM T99041 CS5X9L 46917048 IC50 > 100000 nM T99041 CZP24U 46917049 IC50 = 570 nM T99041 COY5T4 46937042 IC50 = 19 nM T99041 CGMJ52 46938499 IC50 > 100000 nM T99041 C5RAS7 46938602 IC50 > 100000 nM T99041 C3B1LX 46938704 IC50 > 100000 nM T99041 C5TU1F 46938705 IC50 > 100000 nM T99041 CAGP83 46938706 IC50 > 100000 nM T99041 CP9V8Q 46938799 IC50 > 100000 nM T99041 CAB2H9 46938802 IC50 > 100000 nM T99041 C80RAT 47370344 IC50 > 100000 nM T99041 CR5X3K 49785099 IC50 = 0.33 nM T99041 C2HU0V 49785100 IC50 = 1.72 nM T99041 CX7M2K 49785101 IC50 = 0.87 nM T99041 C3XCV4 49785102 IC50 = 1.32 nM T99041 CC8Z5M 49795916 IC50 = 500 nM T99041 CI6U4M 49795917 IC50 = 700 nM T99041 C7HV2K 49795919 IC50 = 2300 nM T99041 CHE51J 49795928 IC50 = 5000 nM T99041 CI6QC3 49795929 IC50 = 800 nM T99041 C8GIY2 49795930 IC50 = 9100000 nM T99041 C2Y5FT 49795931 IC50 = 36 nM T99041 CS1TY7 49795932 IC50 = 23 nM T99041 CUW13V 49795933 IC50 = 47000 nM T99041 CZNL37 49795934 IC50 = 1800000 nM T99041 CGQC72 49795935 IC50 = 31000 nM T99041 CK72BR 49795936 IC50 = 22000 nM T99041 CNB64H 49795937 IC50 = 30 nM T99041 CE2P1Y 49795938 IC50 = 190000 nM T99041 C2TY4D 49795939 IC50 > 10000 nM T99041 COHI43 49795940 IC50 = 400 nM T99041 CDI04P 49795942 IC50 = 1400 nM T99041 CKF3D9 49795943 IC50 = 5000 nM T99041 C95AGZ 49795944 IC50 = 600 nM T99041 CT3XF0 49795948 IC50 = 16 nM T99041 C5RP2S 49796932 IC50 = 510 nM T99041 CZ7A9E 49796933 IC50 = 87 nM T99041 C8D7IG 49796934 IC50 = 539 nM T99041 CBX38D 49796935 IC50 = 1200 nM T99041 CC74RX 49796936 IC50 = 161 nM T99041 CLBU64 49796937 IC50 = 54 nM T99041 C5RF0Y 49796938 IC50 = 7200 nM T99041 CE0C3Y 49796939 IC50 = 75 nM T99041 CI4ZE6 49796940 IC50 = 37 nM T99041 CA54TF 49796941 IC50 = 0.3 nM T99041 CBD8K2 49796942 IC50 = 39 nM T99041 CD21SQ 49796943 IC50 = 170 nM T99041 CODZ18 49796944 IC50 = 118 nM T99041 CI25XP 49796945 IC50 = 721 nM T99041 CF65YQ 49796946 IC50 = 1640 nM T99041 C32MAO 49796947 IC50 = 10 nM T99041 CHJ76U 49796948 IC50 = 3.7 nM T99041 CU25OB 49796949 IC50 = 5.1 nM T99041 C1ZJS7 49796950 IC50 = 4200 nM T99041 C8GWI5 49796951 IC50 = 1.8 nM T99041 CH2W5L 49796952 IC50 = 18 nM T99041 C8WYA5 49796953 IC50 = 0.48 nM T99041 C0P6JR 49796954 IC50 = 1.6 nM T99041 CQH86V 49796955 IC50 = 8.2 nM T99041 C08NMS 49796956 IC50 = 0.83 nM T99041 CR63MS 49796957 IC50 = 18 nM T99041 CJ5FR6 49796958 IC50 = 7.1 nM T99041 C7IBX0 49796959 IC50 = 3300 nM T99041 CU83MS 49796960 IC50 = 12 nM T99041 CQ5YV7 49796961 IC50 = 13 nM T99041 C1T9ON 49796962 IC50 = 3600 nM T99041 C1ZVH6 49796963 IC50 = 82 nM T99041 CB26OQ 49796964 IC50 = 1200 nM T99041 C0NO8F 49796965 IC50 = 9.5 nM T99041 C69JQC 49796966 IC50 = 33 nM T99041 C01RDX 49796967 IC50 = 1.7 nM T99041 C2SXO4 49796968 IC50 = 1.6 nM T99041 C7SH5C 49796969 IC50 = 12 nM T99041 C7K3HC 49796970 IC50 = 295 nM T99041 CBMV50 49796972 IC50 = 64 nM T99041 C8IL0K 49796973 IC50 = 980 nM T99041 CA90LB 49796974 IC50 = 1600 nM T99041 C07DHG 49796977 IC50 = 3500 nM T99041 CAS2P4 49796982 IC50 = 220 nM T99041 CG79KT 49796985 IC50 = 390 nM T99041 C4D8RE 49796990 IC50 = 6.6 nM T99041 CUKB68 49796994 IC50 = 550 nM T99041 CUR9B0 49796995 IC50 = 9.2 nM T99041 CWHO58 49796998 IC50 = 45 nM T99041 CX74RG 49796999 IC50 = 12 nM T99041 C20MAQ 49797000 IC50 = 13 nM T99041 CD67OX 49797001 IC50 = 192 nM T99041 C9LEF5 49797002 IC50 = 9.1 nM T99041 CO2AX9 49797003 IC50 = 3.3 nM T99041 CEM61W 49797006 IC50 = 520 nM T99041 C7Y0JL 49797007 IC50 = 59 nM T99041 CW45IK 49797008 IC50 = 37 nM T99041 C79JUI 49797011 IC50 = 67 nM T99041 CVAK94 49797012 IC50 = 29 nM T99041 CUK5J1 49797013 IC50 = 43 nM T99041 C4ZK5C 49797014 IC50 = 2.2 nM T99041 C1PV8J 49797015 IC50 = 30 nM T99041 C9YEU6 49797016 IC50 = 17 nM T99041 CZD4S2 49797017 IC50 = 99 nM T99041 CKY80F 49797018 IC50 = 11 nM T99041 CS0D8Q 49797021 IC50 = 27 nM T99041 C3GF4M 49797022 IC50 = 100 nM T99041 C8XZT9 49797023 IC50 = 71 nM T99041 C5H2AS 49797024 IC50 = 94 nM T99041 C4P0VW 49797025 IC50 = 20 nM T99041 CVY8M1 49797028 IC50 = 110 nM T99041 CM59HB 49797029 IC50 = 230 nM T99041 CH7Y1J 49797030 IC50 = 44 nM T99041 CX18HI 49797031 IC50 = 21 nM T99041 CUM28Z 49797035 IC50 = 110 nM T99041 COS23G 49797036 IC50 = 7.5 nM T99041 C2TSG6 49797038 IC50 = 56 nM T99041 C7BI3W 49797039 IC50 = 21 nM T99041 C71THK 49797040 IC50 = 1100 nM T99041 C0SG5O 49797041 IC50 = 7900 nM T99041 CM37VB 49797042 IC50 = 170 nM T99041 C51NUG 49797043 IC50 = 480 nM T99041 C65WXC 49797044 IC50 = 600 nM T99041 CHTO37 49797045 IC50 = 2000 nM T99041 CA8R5K 49797046 IC50 = 3700 nM T99041 CLAR35 49797047 IC50 = 250 nM T99041 C9OCZ3 49797048 IC50 = 54000 nM T99041 C49RUW 49797049 IC50 = 1100 nM T99041 C4EHT7 49797050 IC50 = 3700 nM T99041 CW6G5R 49797051 IC50 = 2800 nM T99041 CUK6G0 49797052 IC50 = 120 nM T99041 CJ1FE2 49797053 IC50 = 280 nM T99041 CKJO08 49797054 IC50 = 4200 nM T99041 C70KVU 49797055 IC50 = 3600 nM T99041 CP59BI 49797056 IC50 = 360 nM T99041 CEDL61 49797057 IC50 = 770 nM T99041 C5J2LV 49797058 IC50 = 1400 nM T99041 CEI20Q 49797059 IC50 = 1100 nM T99041 C7B5DY 49797060 IC50 = 6 nM T99041 C5B1RM 49797061 IC50 = 100 nM T99041 C40HJC 49797062 IC50 = 240 nM T99041 CL3P4H 49797063 IC50 = 98 nM T99041 CPC76U 49797064 IC50 = 140 nM T99041 C5F4JN 49797065 IC50 = 580 nM T99041 C86HND 49797066 IC50 = 130 nM T99041 C8E4XD 49797067 IC50 = 1500 nM T99041 CHO1U0 49797068 IC50 = 100 nM T99041 CO1TW7 49797069 IC50 = 69 nM T99041 CAD6W1 49797071 IC50 = 110 nM T99041 CQYU80 49797072 IC50 = 110 nM T99041 CEZ38H 49797073 IC50 = 110 nM T99041 C0CEU7 49797074 IC50 = 140 nM T99041 C72JXY 49797075 IC50 = 27 nM T99041 COA41Q 49797076 IC50 = 510 nM T99041 CPQ3Z2 49797077 IC50 = 140 nM T99041 C1WI0D 49797078 IC50 = 60 nM T99041 C4D8XP 49797079 IC50 = 390 nM T99041 CQG4J6 49797080 IC50 = 130 nM T99041 CKM9S4 49797081 IC50 = 75 nM T99041 C3JRW0 49797082 IC50 = 370 nM T99041 C27IEB 49797083 IC50 = 150 nM T99041 C0JUL3 49797084 IC50 = 110 nM T99041 C85DOL 49797085 IC50 = 110 nM T99041 CEGO30 49797086 IC50 = 150 nM T99041 C2TC3I 49797087 IC50 = 440 nM T99041 C04JWY 49797088 IC50 = 240 nM T99041 CA2U4Y 49797089 IC50 = 56 nM T99041 CFT46J 49797090 IC50 = 37 nM T99041 C35TFW 49797091 IC50 = 86 nM T99041 CRL7Z5 49797092 IC50 = 710 nM T99041 CYU74X 49797093 IC50 = 420 nM T99041 C2O3SG 49797094 IC50 = 150 nM T99041 CFL3O2 49797106 IC50 = 48 nM T99041 CF4NR7 49797107 IC50 = 26 nM T99041 CV9QW6 49797108 IC50 = 31 nM T99041 CJZA65 49797109 IC50 = 1100 nM T99041 CBS36X 49797110 IC50 = 38 nM T99041 C0STP5 49797111 IC50 = 29 nM T99041 C7KV5R 49797112 IC50 = 320 nM T99041 CJPX53 49797113 IC50 = 570 nM T99041 C2OI0Y 49797114 IC50 = 25 nM T99041 CW20FJ 49797115 IC50 = 34 nM T99041 C9P6VU 49797116 IC50 = 49 nM T99041 C67SIA 49797117 IC50 = 74 nM T99041 CCI8Y0 49797118 IC50 = 67 nM T99041 CE10UF 49797119 IC50 = 37 nM T99041 CLH0V3 49797120 IC50 = 120 nM T99041 C2N8WX 49797121 IC50 = 26 nM T99041 CNCE06 49797122 IC50 = 90 nM T99041 C76UAB 49797123 IC50 = 69 nM T99041 CHWT89 49797124 IC50 = 92 nM T99041 C1Z6NE 49797125 IC50 = 61 nM T99041 C25MQG 49797126 IC50 = 229 nM T99041 COL54B 49797127 IC50 = 117 nM T99041 C5OUQ3 49797128 IC50 = 52 nM T99041 C3NMI8 49797173 Ki = 12 nM T99041 C1E3YB 49797174 Ki = 6 nM T99041 CVD0I1 49797175 Ki = 3.6 nM T99041 CH02OC 49797176 Ki = 4.7 nM T99041 CY1OJ5 49797177 Ki = 1.3 nM T99041 CL8TW4 49797178 Ki < 140 nM T99041 C25ZSD 49797191 IC50 = 203 nM T99041 C0OJX9 49797192 IC50 = 8 nM T99041 C7GZ4B 49797193 IC50 = 19 nM T99041 CVT2E5 49797194 IC50 = 40 nM T99041 C75MGE 49797195 IC50 = 13 nM T99041 CVS70C 49797196 IC50 = 13 nM T99041 C42QPW 49797197 IC50 = 70 nM T99041 C6ZGL5 49797198 IC50 = 52 nM T99041 C1B5NH 49797199 IC50 = 31 nM T99041 CGQN24 49797200 IC50 = 560 nM T99041 CS2AI5 49797201 IC50 = 1210 nM T99041 CM7RE3 49797202 IC50 = 1830 nM T99041 CGM9E7 49797203 IC50 = 3050 nM T99041 COU0I6 49797204 IC50 = 19 nM T99041 C3XML2 49797205 IC50 = 19 nM T99041 CP0O2F 49797223 IC50 = 210 nM T99041 CTH7I8 49797224 IC50 = 58 nM T99041 CG9P7O 49797225 IC50 = 144 nM T99041 C3A2QK 49797226 IC50 = 125 nM T99041 C4NOK2 49797227 IC50 = 111 nM T99041 CB13PO 49797228 IC50 = 67 nM T99041 C47VOG 49797229 IC50 = 463 nM T99041 CD2CL1 49797230 IC50 = 650 nM T99041 C0LK6B 49797231 IC50 = 14 nM T99041 CON0A6 49797232 IC50 = 37 nM T99041 C4AVU3 49797233 IC50 = 90 nM T99041 CQ93MI 49797234 IC50 = 82 nM T99041 CO2JV8 49797235 IC50 = 63 nM T99041 C27LDC 49797236 IC50 = 54 nM T99041 CA5GM6 49797237 IC50 = 3700 nM T99041 CT8PW1 49797238 IC50 = 7 nM T99041 CJQ38S 49797239 IC50 = 12 nM T99041 CT65MR 49797240 IC50 = 130 nM T99041 C08IFZ 49797241 IC50 = 43 nM T99041 CA4E8M 49797242 IC50 = 13 nM T99041 CN8FR2 49797243 IC50 = 22 nM T99041 C37MDP 49797244 IC50 = 5 nM T99041 CM41RN 49797245 IC50 = 2 nM T99041 C59JEK 49797246 IC50 = 8 nM T99041 CUMH43 49797248 IC50 = 8 nM T99041 CM59PE 49797249 IC50 = 5 nM T99041 CN5K1S 49797250 IC50 = 31 nM T99041 CT5HY0 49797251 IC50 = 6 nM T99041 C0E5PY 49797252 IC50 = 9 nM T99041 C3E5JB 49797253 IC50 = 16 nM T99041 CA8P5N 49797344 IC50 = 870 nM T99041 CJL2B8 49797345 IC50 = 430 nM T99041 CT79YI 49797346 IC50 = 25 nM T99041 C93VJO 49797347 IC50 = 160 nM T99041 CDI52A 49797348 IC50 = 300 nM T99041 C7ATK9 49797349 IC50 = 160 nM T99041 C2Y3DS 49797350 IC50 = 600 nM T99041 CA4CE3 49797351 IC50 = 150 nM T99041 C3A8YT 49797352 IC50 = 210 nM T99041 C1Z8HB 49797353 IC50 = 48 nM T99041 CC0T8H 49797354 IC50 = 330 nM T99041 C92QND 49797355 IC50 = 1490 nM T99041 C2HPE8 49797356 IC50 = 1280 nM T99041 C9UXH2 49797357 IC50 = 440 nM T99041 CTYO37 49797358 IC50 = 24 nM T99041 C1K4FR 49797359 IC50 = 22 nM T99041 CJ2D0P 49797360 IC50 = 74 nM T99041 CA3Q2W 49797361 IC50 = 29 nM T99041 CNMF62 49797362 IC50 = 21 nM T99041 C3HU6X 49797446 IC50 = 1490 nM T99041 C3U1KQ 49797450 IC50 = 525 nM T99041 C76KMB 49797451 IC50 = 17 nM T99041 C02MPV 49797452 IC50 = 122 nM T99041 CLVF17 49797501 IC50 = 9 nM T99041 CR0AK2 49797502 IC50 = 6 nM T99041 CM1Y7K 49797503 IC50 = 7 nM T99041 CUSI73 49797504 IC50 = 10 nM T99041 CJ0DX6 49797505 IC50 = 22 nM T99041 C2A7LE 49797506 IC50 = 7 nM T99041 CU4M3T 49797507 IC50 = 15 nM T99041 C8GCS5 49797508 IC50 = 17 nM T99041 CTP9L2 49797509 IC50 = 31 nM T99041 CT76PM 49797510 IC50 = 8 nM T99041 C4K0QT 49797511 IC50 = 19 nM T99041 CLHB50 49797512 IC50 = 37 nM T99041 CC56FE 49797513 IC50 = 11 nM T99041 C4T6AB 49797514 IC50 = 8 nM T99041 C41VHF 49797515 IC50 = 31 nM T99041 CBD9H2 49797516 IC50 = 12 nM T99041 CAOC90 49797517 IC50 = 31 nM T99041 C0F5QX 49797518 IC50 = 12 nM T99041 C7T5XW 49797519 IC50 = 16 nM T99041 CM6SF5 49797520 IC50 = 25 nM T99041 CQZN45 49797521 IC50 = 14 nM T99041 CG64BU 49797522 IC50 = 13 nM T99041 C5G3MA 49797524 IC50 = 5 nM T99041 CO42DE 49797525 IC50 = 35 nM T99041 C5L1EP 49797526 IC50 = 40 nM T99041 CTWR80 49797527 IC50 = 6 nM T99041 CPIC42 49797528 IC50 = 7 nM T99041 C5N1ZB 49797529 IC50 = 5 nM T99041 CU72EZ 49797596 IC50 = 17 nM T99041 C6AZ2C 49797599 IC50 = 52 nM T99041 CR86PO 49797604 IC50 = 22 nM T99041 C6DJX7 49797605 IC50 = 4.2 nM T99041 CK3ZI1 49797607 IC50 = 7.1 nM T99041 C7AD0C 49797610 IC50 = 53 nM T99041 C4XHO5 49797612 IC50 = 8 nM T99041 C7VL5U 49797614 IC50 = 28 nM T99041 CY09JE 49797615 IC50 = 47 nM T99041 C1ZLF0 49797616 IC50 = 13 nM T99041 CN48OE 49797627 IC50 = 77 nM T99041 CV6I0O 49797630 IC50 = 14 nM T99041 CAG1U7 49797631 IC50 = 56 nM T99041 C8JNU1 49797636 IC50 = 68 nM T99041 C0DN5G 49797642 IC50 = 47 nM T99041 CJVS96 49797644 IC50 = 18 nM T99041 CBRT78 49797650 IC50 = 8.6 nM T99041 CZW93Y 49797653 IC50 = 30 nM T99041 COM5Q7 49836030 IC50 = 27 nM T99041 CKZJ30 49837952 IC50 = 16 nM T99041 CXR05H 49837954 IC50 = 11 nM T99041 C4QSP1 49837961 IC50 = 10 nM T99041 C1WSF0 49843627 IC50 = 300 nM T99041 C31PHS 49843629 IC50 = 101 nM T99041 CDAK59 49843631 IC50 = 124 nM T99041 CSWR53 49845007 IC50 = 2300 nM T99041 C02RWO 49845009 IC50 = 1060 nM T99041 CG5O9N 49845011 IC50 = 1240 nM T99041 C9ST1E 49845161 IC50 = 460 nM T99041 C64NVQ 49845166 IC50 = 1236 nM T99041 C3CVF2 49845349 IC50 = 360 nM T99041 CTDR85 49862539 Ki = 73 nM T99041 CT8Q9N 49862713 Ki = 73 nM T99041 C0OB8C 49862714 Ki = 50 nM T99041 CJ58AG 49862715 Ki = 50 nM T99041 C42TSR 49862716 Ki = 31 nM T99041 CPU7F6 49862790 Ki = 29 nM T99041 C4FZY2 49862791 Ki = 442 nM T99041 CF40YM 49862792 Ki = 106 nM T99041 CK0GC5 49864113 Ki = 5.4 nM T99041 CK1CD3 50925423 IC50 = 23 nM T99041 C8XA7H 50942035 IC50 = 13 nM T99041 CFT4L5 50970490 IC50 = 93 nM T99041 C7T6PI 50994092 IC50 = 1.1 nM T99041 C67CTP 51032641 IC50 = 88.82 nM T99041 C1ECS9 51050448 IC50 = 66 nM T99041 CL4S9Y 51050450 IC50 = 39 nM T99041 CWZ76P 51050544 IC50 = 23 nM T99041 CT3D7J 51050546 IC50 = 8.7 nM T99041 C5O1PJ 51050548 IC50 = 9.6 nM T99041 CR6ZG8 51050550 IC50 = 6.6 nM T99041 CY3W8O 51051127 IC50 = 57 nM T99041 C2GNK6 51051129 IC50 = 58 nM T99041 CLU39H 51051131 IC50 = 18 nM T99041 C5PRF8 51051132 IC50 = 18 nM T99041 CYF04M 51051134 IC50 = 5.7 nM T99041 CPCY75 51051136 IC50 = 4.4 nM T99041 C7JM3I 51051236 IC50 = 19 nM T99041 CZ5HJ0 51051238 IC50 = 4.6 nM T99041 C1OUG5 51051240 IC50 = 2.5 nM T99041 C6GAP9 51051329 IC50 = 20 nM T99041 C9KPJ6 51051331 IC50 = 10 nM T99041 C85CEJ 51346970 IC50 = 55 nM T99041 C4PFT3 51346971 IC50 = 94 nM T99041 CLG9I5 51355035 IC50 = 89.5 nM T99041 CLND76 51356956 IC50 = 44 nM T99041 CH92AI 51356957 IC50 = 80 nM T99041 CH89VX 51356958 IC50 = 686 nM T99041 C5D4HV 51356959 IC50 = 674 nM T99041 C03ROM 51356960 IC50 < 50000 nM T99041 C8WOG2 51356962 IC50 = 674 nM T99041 CJ0Q4A 52918281 IC50 = 50.66 nM T99041 C4VC2U 52942435 IC50 = 87 nM T99041 C2B6EX 52943488 Ki = 11 nM T99041 CGOM96 52943515 IC50 = 114 nM T99041 C56CXU 52943631 IC50 = 151 nM T99041 CHD7O6 52943758 IC50 = 13 nM T99041 C4I6ML 52944843 IC50 = 23 nM T99041 C57XSM 52944845 IC50 = 122 nM T99041 CT6SQ3 52944941 IC50 = 28 nM T99041 C7RJM9 52945660 IC50 = 10 nM T99041 C9OAF1 52946149 IC50 = 1.8 nM T99041 CBVC96 52946447 IC50 = 10 nM T99041 CC56BV 52946866 IC50 > 100000 nM T99041 CC7N8S 52948914 IC50 = 36 nM T99041 C4LVO6 52948971 IC50 = 12 nM T99041 CTU0J1 52949742 IC50 = 103 nM T99041 CD4HQ1 53233695 IC50 = 3100 nM T99041 C89KWN 53233798 IC50 = 4000 nM T99041 CEFX05 53311069 IC50 = 1100 nM T99041 CQL50R 53311070 IC50 > 100000 nM T99041 C1Q4WK 53311071 IC50 = 20000 nM T99041 C67LHZ 53311072 IC50 = 530 nM T99041 CQ0ZJ2 53311073 IC50 = 5200 nM T99041 C7PMY1 53311074 IC50 = 38000 nM T99041 CWN9H7 53311140 IC50 = 100 nM T99041 CAL51C 53311141 IC50 = 16000 nM T99041 C2SXV0 53311142 IC50 = 88000 nM T99041 C7AEF8 53311143 IC50 > 100000 nM T99041 C5IOZ6 53311144 IC50 = 3400 nM T99041 CVR4H3 53311222 IC50 = 430 nM T99041 CNX08H 53311223 IC50 = 110 nM T99041 CET6W5 53311225 IC50 = 2500 nM T99041 C3RZS4 53311226 IC50 = 480 nM T99041 CHR17Y 53311227 IC50 = 13 nM T99041 C3HGW8 53312238 IC50 > 100000 nM T99041 CM03UX 53312239 IC50 > 100000 nM T99041 C9K4CZ 53312243 IC50 > 100000 nM T99041 CU4BS2 53312323 IC50 = 23000 nM T99041 CF5I6O 53312326 IC50 = 22 nM T99041 C6PSL2 53312327 IC50 > 100000 nM T99041 C0WYS5 53312328 IC50 = 45 nM T99041 CI0Z2A 53317343 IC50 > 50000 nM T99041 CLZ1M4 53317345 IC50 > 50000 nM T99041 CO3SY5 53317346 IC50 > 50000 nM T99041 C4M7TX 53317347 IC50 > 50000 nM T99041 C37HQG 53317348 IC50 > 50000 nM T99041 CYC69Q 53317564 IC50 = 85 nM T99041 C0QOV9 53317565 IC50 = 180 nM T99041 CURC70 53317566 IC50 = 400 nM T99041 C3ZK1W 53317575 IC50 = 120 nM T99041 CBQ0J7 53317579 IC50 = 280 nM T99041 CIY9F7 53317580 IC50 = 57 nM T99041 C5DMS9 53317581 IC50 = 450 nM T99041 C1XD9W 53317582 IC50 = 82 nM T99041 CR0O8T 53317583 IC50 = 18 nM T99041 CHW98L 53317619 IC50 = 13 nM T99041 C9AB1E 53317627 IC50 = 488 nM T99041 C0XQ2B 53318462 IC50 = 22.53 nM T99041 CJO28A 53318492 IC50 = 29.92 nM T99041 C45YDV 53318494 IC50 = 52.34 nM T99041 C6H4ZL 53318496 IC50 = 30.03 nM T99041 CYBP96 53318498 IC50 = 36.43 nM T99041 C9GLH7 53318841 IC50 = 84 nM T99041 C06TDE 53318842 IC50 = 150 nM T99041 C73TER 53318856 IC50 = 110 nM T99041 CC56NE 53318863 IC50 = 110 nM T99041 C4UJI8 53318864 IC50 = 310 nM T99041 C8CZ2A 53318865 IC50 = 110 nM T99041 CLVY47 53318866 IC50 = 51 nM T99041 CQC8N4 53318918 IC50 = 80 nM T99041 C7P2UE 53318921 IC50 = 1400 nM T99041 CP67YM 53318983 IC50 > 50000 nM T99041 C6SJ4Z 53318987 IC50 = 74 nM T99041 CM7S5W 53319067 IC50 = 110 nM T99041 C85NSB 53319824 IC50 = 37.54 nM T99041 CTW2R8 53319826 IC50 = 46.89 nM T99041 CW83TR 53319828 IC50 = 15.8 nM T99041 CC59LI 53319949 IC50 > 50000 nM T99041 CNW4K5 53319950 IC50 > 50000 nM T99041 CQK53D 53319951 IC50 > 50000 nM T99041 CD9LA8 53320113 IC50 > 50000 nM T99041 C1X3NE 53320178 IC50 = 120 nM T99041 C1P8BK 53320179 IC50 = 110 nM T99041 C50UBZ 53320180 IC50 = 140 nM T99041 C2JTR7 53320181 IC50 = 260 nM T99041 C0TYJ5 53320182 IC50 = 77 nM T99041 C7RSX2 53320183 IC50 = 72 nM T99041 CJU34O 53320232 IC50 = 19 nM T99041 C8ML9Y 53321113 IC50 = 45.2 nM T99041 CF0B3T 53321115 IC50 = 46.61 nM T99041 CEO6M2 53321117 IC50 = 22.76 nM T99041 CFPY75 53321119 IC50 = 17.83 nM T99041 CXZ47P 53321201 IC50 < 50000 nM T99041 CJ2V8E 53321202 IC50 = 937 nM T99041 CGVE79 53321203 IC50 < 50000 nM T99041 CP12HY 53321204 IC50 < 50000 nM T99041 C0XLS2 53321252 IC50 < 50000 nM T99041 CNT89R 53321253 IC50 > 50000 nM T99041 CO58YD 53321254 IC50 > 50000 nM T99041 C9XGE4 53321472 IC50 = 140 nM T99041 CY0ZV9 53321485 IC50 = 170 nM T99041 CK0OB2 53321486 IC50 = 38 nM T99041 CNK34J 53321487 IC50 = 260 nM T99041 C7EO3D 53321495 IC50 = 140 nM T99041 C3M7PQ 53321496 IC50 = 850 nM T99041 C0NUQ7 53321497 IC50 = 330 nM T99041 C31DSJ 53321498 IC50 = 450 nM T99041 C2ZKV9 53321499 IC50 = 71 nM T99041 CGA05O 53321545 IC50 = 216 nM T99041 CAU2F0 53321549 IC50 = 12 nM T99041 CB76JK 53321550 IC50 = 59 nM T99041 C50RJL 53321566 IC50 = 13 nM T99041 C3QT0R 53321621 IC50 = 140 nM T99041 CF2GQ1 53321670 IC50 = 22 nM T99041 C4UA2C 53322441 IC50 = 12.4 nM T99041 CF5M0P 53322443 IC50 = 33.17 nM T99041 CQK38R 53322445 IC50 = 33.25 nM T99041 C3OTG6 53322447 IC50 = 47.27 nM T99041 CKT3E2 53322456 IC50 = 77.06 nM T99041 CR9TY2 53322529 IC50 > 50000 nM T99041 C56URQ 53322530 IC50 < 50000 nM T99041 C1ZIS9 53322575 IC50 > 50000 nM T99041 C2MA6T 53322742 IC50 > 50000 nM T99041 CXIS21 53322758 IC50 = 730 nM T99041 CY71QL 53322814 IC50 = 130 nM T99041 CLU96Y 53322820 IC50 = 270 nM T99041 C8YVF1 53322821 IC50 = 290 nM T99041 C4QS6V 53322822 IC50 = 220 nM T99041 C62JTB 53322823 IC50 = 710 nM T99041 CT14FU 53322824 IC50 = 690 nM T99041 CXJ1F8 53322825 IC50 = 670 nM T99041 C3K1VY 53322826 IC50 = 21 nM T99041 CC09IP 53322885 IC50 = 41 nM T99041 C9N6HK 53322952 IC50 = 70 nM T99041 C7NUF3 53323807 IC50 = 28.6 nM T99041 C3QGT8 53323865 IC50 < 50000 nM T99041 C0FOV2 53323866 IC50 < 50000 nM T99041 CZ4I5J 53323915 IC50 < 50000 nM T99041 C4E8OK 53323916 IC50 > 50000 nM T99041 CB7HG9 53323917 IC50 > 50000 nM T99041 C9LU8M 53324129 IC50 = 99 nM T99041 CCY7M0 53324130 IC50 = 130 nM T99041 C4F1QK 53324142 IC50 = 500 nM T99041 CZN71C 53324143 IC50 = 670 nM T99041 CG83JZ 53324144 IC50 = 140 nM T99041 CE8J1D 53324145 IC50 = 140 nM T99041 C0Y3AC 53324153 IC50 = 120 nM T99041 C9O1IW 53324154 IC50 = 910 nM T99041 CTW5G0 53324155 IC50 = 130 nM T99041 C2DPZ0 53324156 IC50 = 54 nM T99041 C9A4JG 53324203 IC50 = 28 nM T99041 CPCE78 53324209 IC50 = 47 nM T99041 C6CJ0H 53324210 IC50 = 1.6 nM T99041 CL5Z8N 53324211 IC50 = 39 nM T99041 CV7UM8 53324212 IC50 = 37 nM T99041 C98EJV 53324213 IC50 = 13 nM T99041 CSN28M 53324293 IC50 = 2400 nM T99041 C2FRA0 53324311 IC50 > 50000 nM T99041 CDW31Y 53325018 IC50 < 50000 nM T99041 C76TDZ 53325194 IC50 < 50000 nM T99041 CJWL87 53325195 IC50 > 50000 nM T99041 CBT0Z8 53325196 IC50 > 50000 nM T99041 C2N5BX 53325197 IC50 > 50000 nM T99041 CF65NE 53325325 IC50 = 77 nM T99041 C25OJW 53325399 IC50 = 430 nM T99041 CXW5O9 53325446 IC50 = 280 nM T99041 C1SO0C 53325447 IC50 = 570 nM T99041 C1S3WB 53325453 IC50 = 200 nM T99041 C2KFW6 53325454 IC50 = 75 nM T99041 C4ZFR5 53325455 IC50 = 78 nM T99041 CPS51R 53325503 IC50 = 153 nM T99041 CW8TM9 53325504 IC50 = 26 nM T99041 CCOQ72 53325553 IC50 = 26.17 nM T99041 C5UB1G 53325568 IC50 < 50000 nM T99041 C1Z4RT 53326344 IC50 = 15.09 nM T99041 CX6Q3E 53326370 IC50 = 75.35 nM T99041 C30OEU 53326372 IC50 = 26.64 nM T99041 CL7T1U 53326374 IC50 = 33.78 nM T99041 CJP5V7 53326443 IC50 < 50000 nM T99041 C65JNF 53326490 IC50 > 50000 nM T99041 CYIA49 53326515 IC50 = 2.8 nM T99041 CV0H8P 53326691 IC50 = 110 nM T99041 C3ZWN6 53326704 IC50 = 100 nM T99041 C73SKG 53326705 IC50 = 1300 nM T99041 CG9V4W 53326706 IC50 = 110 nM T99041 C5K8CP 53326713 IC50 = 100 nM T99041 CHCE65 53326766 IC50 = 51 nM T99041 C4LCU1 53326767 IC50 = 1.2 nM T99041 C9UBW8 53326841 IC50 > 50000 nM T99041 C1HYV2 53326876 IC50 > 50000 nM T99041 CN12AO 53353383 IC50 = 255 nM T99041 C51GUC 53354365 IC50 = 67 nM T99041 CRJ5P9 53354369 IC50 = 102 nM T99041 C4G2HT 53354470 IC50 = 57 nM T99041 CUC1N3 53356519 Ki = 0.37 nM T99041 CSD1Q4 53357353 IC50 = 1.1 nM T99041 C5P9VZ 53465973 IC50 > 100000 nM T99041 C7OBF2 53465974 IC50 > 100000 nM T99041 CF5YJ8 53465975 IC50 > 100000 nM T99041 C5XER7 53466046 IC50 > 100000 nM T99041 CJ9T8M 53466047 IC50 > 50000 nM T99041 CP1CL8 53466049 IC50 > 100000 nM T99041 CPSQ16 53466050 IC50 > 100000 nM T99041 C4UC1P 53466119 IC50 > 100000 nM T99041 C59SML 53466121 IC50 > 100000 nM T99041 C7JPY2 53466122 IC50 > 100000 nM T99041 CYZK63 53466123 IC50 > 50000 nM T99041 CVJ0D5 53466193 IC50 > 100000 nM T99041 C2XE8Y 53466195 IC50 > 100000 nM T99041 C0P2YE 53466196 IC50 > 100000 nM T99041 CPA0K4 53466271 IC50 > 100000 nM T99041 CYG36O 53466361 IC50 = 17700 nM T99041 C5J9EB 53770701 IC50 = 510 nM T99041 CEK45S 54294055 IC50 = 87000 nM T99041 CRL42P 54573912 IC50 = 400 nM T99041 CUZS62 54580221 IC50 = 19 nM T99041 CG3S0X 54580222 IC50 = 0.7 nM T99041 CAQ8U7 54580310 IC50 = 21300 nM T99041 CX6K2C 54580311 IC50 = 26200 nM T99041 CS21IF 54580575 IC50 = 44.8 nM T99041 COZ98J 54580576 IC50 = 116 nM T99041 C2TSH1 54580577 IC50 = 54.1 nM T99041 CZL0N3 54580578 IC50 = 30.8 nM T99041 CNAQ35 54580579 IC50 = 7.4 nM T99041 CT24DU 54581222 IC50 = 7 nM T99041 CABF19 54581317 IC50 = 32700 nM T99041 C9JBG4 54581584 IC50 = 26.7 nM T99041 CJZ4S8 54582330 IC50 = 29100 nM T99041 C4L9SF 54582574 IC50 = 38.5 nM T99041 C0LQ9Z 54582575 IC50 = 13.7 nM T99041 CG84BL 54582898 IC50 = 12 nM T99041 CE5X6H 54583545 IC50 = 33.9 nM T99041 CB52YA 54583546 IC50 = 12 nM T99041 CST5M7 54584528 IC50 = 311 nM T99041 CV10YB 54585462 IC50 = 42.7 nM T99041 CG6M8J 54585463 IC50 = 38.9 nM T99041 CLCU50 54585464 IC50 = 1.3 nM T99041 CPWB63 54586434 IC50 = 50.7 nM T99041 C4G2PK 54586435 IC50 = 29 nM T99041 C71GKO 54586787 IC50 = 3 nM T99041 C4B2EW 54587461 IC50 = 92.6 nM T99041 C7VL9M 54587462 IC50 = 48.9 nM T99041 C04FAR 54587463 IC50 = 33.8 nM T99041 CQH56N 54698732 IC50 = 730 nM T99041 CY0ZH5 54698792 IC50 = 2950 nM T99041 C5UW0D 56652661 IC50 = 45 nM T99041 CMT0J9 56656630 IC50 = 133.6 nM T99041 C1QX0O 56657809 IC50 = 2 nM T99041 CU74VH 56658024 IC50 > 100000 nM T99041 CF6PV5 56658026 IC50 > 100000 nM T99041 C2KI8Y 56658028 IC50 > 100000 nM T99041 CY4E6U 56658138 IC50 > 100000 nM T99041 C5OT6W 56658248 IC50 = 26 nM T99041 C07KTW 56658249 IC50 > 1000 nM T99041 C1UDJ5 56659853 IC50 = 34 nM T99041 CX31TJ 56661748 IC50 = 0.34 nM T99041 COI5B0 56663604 IC50 = 65.1 nM T99041 C3VIA8 56663606 IC50 = 68.1 nM T99041 CD31AI 56663612 IC50 = 29.3 nM T99041 C52TBZ 56664349 IC50 = 20.4 nM T99041 C1PI4L 56664962 IC50 > 100000 nM T99041 C8GPO1 56665883 IC50 = 190 nM T99041 CA0BO6 56666264 IC50 > 100000 nM T99041 C8F5QV 56666543 IC50 = 4.2 nM T99041 C76MXW 56666747 IC50 = 49 nM T99041 C8DB0L 56670173 IC50 = 57 nM T99041 CJ9Q3V 56670497 IC50 = 47.8 nM T99041 CNL7D4 56671283 IC50 = 68.6 nM T99041 CXH5W7 56671896 IC50 > 100000 nM T99041 CMW3T8 56673186 IC50 > 100000 nM T99041 C1Q4XU 56673980 IC50 = 165.6 nM T99041 CP87EK 56674589 IC50 = 60.1 nM T99041 C2B6PY 56674700 IC50 = 34.8 nM T99041 C3OHT5 56675121 IC50 = 82.4 nM T99041 CBK31U 56675279 IC50 > 100000 nM T99041 CW8KU6 56675536 IC50 > 50000 nM T99041 C7WCK5 56676440 IC50 = 790 nM T99041 CH13RF 56676769 IC50 = 26 nM T99041 CX92YZ 56676772 IC50 = 2.7 nM T99041 CAO6M3 56677318 IC50 = 53.5 nM T99041 CPT94R 56678428 IC50 = 44.5 nM T99041 CN9S8A 56679836 IC50 > 100000 nM T99041 CF08YD 56680615 IC50 = 25.8 nM T99041 CZ1P7K 56851484 IC50 = 72 nM T99041 CU61OI 56851486 IC50 = 94 nM T99041 C9OL5C 56962798 IC50 = 10 nM T99041 CQX8J0 57385070 IC50 = 13.78 nM T99041 CPS89B 57385071 IC50 = 2.64 nM T99041 CNU9C0 57385072 IC50 = 2.34 nM T99041 CG5MT6 57385073 IC50 = 1.4 nM T99041 CQZ09L 57390626 IC50 = 80 nM T99041 CWR4E5 57390923 Ki = 0.55 nM T99041 C0RAD8 57390924 Ki = 0.3 nM T99041 C2AR3V 57391609 IC50 = 5.5 nM T99041 CKPB03 57391802 IC50 = 4 nM T99041 C8SW9E 57391803 IC50 = 10 nM T99041 C5UWC6 57391804 IC50 = 1 nM T99041 C78QEY 57391805 IC50 = 25 nM T99041 CYAQ83 57391806 IC50 = 20 nM T99041 COL58X 57391831 IC50 = 1 nM T99041 C5U6RF 57392407 IC50 = 13 nM T99041 CD0OT2 57392409 IC50 = 15 nM T99041 C4QYJ6 57392724 Ki = 0.27 nM T99041 CKS3X9 57393534 IC50 = 4 nM T99041 CM2EH0 57393535 IC50 = 250 nM T99041 CNP60T 57393564 IC50 = 10 nM T99041 CWDY79 57394441 Ki = 1.5 nM T99041 C5USX7 57395248 IC50 = 0.5 nM T99041 CJ80BU 57395249 IC50 = 1 nM T99041 C27MRL 57395273 IC50 = 20 nM T99041 CX5MG4 57395274 IC50 = 5 nM T99041 C40WGY 57395275 IC50 = 45 nM T99041 CZ23RJ 57395915 IC50 = 32 nM T99041 C8KMS2 57396206 Ki = 0.4 nM T99041 C0P8KM 57397016 IC50 = 2 nM T99041 CE85SV 57397017 IC50 = 2 nM T99041 C0J9MO 57397044 IC50 = 1 nM T99041 CCZ61A 57397045 IC50 = 8 nM T99041 CZJ1P7 57397046 IC50 = 9 nM T99041 C2QL6K 57397702 IC50 = 1.8 nM T99041 CBQ85O 57397704 IC50 = 11 nM T99041 C2ZE3R 57397706 IC50 = 28 nM T99041 CW97SN 57398006 Ki = 0.67 nM T99041 CSU2O9 57398779 IC50 = 2 nM T99041 C01KCU 57399665 Ki = 0.31 nM T99041 CDQ57A 57400458 IC50 = 3 nM T99041 CED9C4 57400459 IC50 = 2 nM T99041 CSEK63 57400487 IC50 = 4 nM T99041 CH6YT2 57400488 IC50 = 3 nM T99041 CX0N7O 57400489 IC50 = 60 nM T99041 C65ZFW 57401128 IC50 = 110 nM T99041 CYX43T 57401419 Ki = 0.29 nM T99041 CV2ME6 57402260 IC50 = 9 nM T99041 CQ1A8P 57402261 IC50 = 2 nM T99041 CW94QA 57402262 IC50 = 10 nM T99041 CMJA69 57402263 IC50 = 5 nM T99041 CV2CF5 57402294 IC50 = 23 nM T99041 C1T0AD 57403169 Ki = 0.43 nM T99041 C12QCM 57403170 Ki = 0.46 nM T99041 CX94UQ 57403171 Ki = 0.26 nM T99041 CX31VN 57403989 IC50 = 7.5 nM T99041 C4E7UI 57404016 IC50 = 2100 nM T99041 C5FHR8 57404017 IC50 = 15 nM T99041 C1L8YD 57404359 IC50 = 1650 nM T99041 C8SX7A 57404360 IC50 = 1100 nM T99041 C0Q1OZ 57404374 IC50 = 350 nM T99041 CXRS60 57406622 IC50 = 10 nM T99041 CNOX18 57406623 IC50 = 43.5 nM T99041 CZS03L 57406803 IC50 = 1.28 nM T99041 C80RBH 57406804 IC50 = 38.6 nM T99041 CMH17V 57406805 IC50 = 1.61 nM T99041 C2EX0S 57406806 IC50 = 19.3 nM T99041 CR6QP4 57406990 IC50 = 32 nM T99041 CFML71 57406991 IC50 = 8.15 nM T99041 C2PX9N 57406992 IC50 = 44.3 nM T99041 CHV47A 57406994 IC50 = 539 nM T99041 C0COE1 57407188 IC50 = 11.2 nM T99041 C5G3KT 57407189 IC50 = 9.31 nM T99041 C8MJK5 57407191 IC50 = 14.1 nM T99041 CVS34M 57407192 IC50 = 29.2 nM T99041 C7AZB3 57407370 IC50 = 82.2 nM T99041 CL0UA1 57525787 IC50 = 0.37 nM T99041 C75MLI 58874215 IC50 = 5.8 nM T99041 C9ZE7J 58874273 IC50 = 0.48 nM T99041 C3TSN9 58874353 IC50 = 14 nM T99041 C4KDJ8 58874386 IC50 = 0.55 nM T99041 COIQ05 58874405 IC50 = 418 nM T99041 C2I4JY 58874420 IC50 = 3.4 nM T99041 C0F5MP 58874435 IC50 = 4.8 nM T99041 CMW4N9 58874436 IC50 = 103 nM T99041 CZ4VD5 60032916 IC50 = 2.3 nM T99041 CI87CZ 61148520 Ki = 880 nM T99041 CAQ1O3 61148706 IC50 = 3.4 nM T99041 C68SUW 61174564 IC50 = 6.93 nM T99041 CXG48F 66545741 IC50 = 5.6 nM T99041 C2YPI7 66559296 IC50 = 0.61 nM T99041 CO2H1S 66559297 IC50 = 1.6 nM T99041 CRI16X 66559298 IC50 = 0.8 nM T99041 C5CX6V 66559299 IC50 = 0.59 nM T99041 CT15QA 66559300 IC50 = 0.39 nM T99041 CX48AY 66559301 IC50 = 1.2 nM T99041 CO0JP1 66559376 IC50 = 0.5 nM T99041 C2W0LI 66559377 IC50 = 0.55 nM T99041 C0NT6U 66559378 IC50 = 0.42 nM T99041 CG6EY9 66560524 IC50 = 0.61 nM T99041 CQMO80 66560608 IC50 = 0.73 nM T99041 CN4RL2 66560609 IC50 = 0.51 nM T99041 CS30FN 66560610 IC50 = 2.2 nM T99041 CZ4OU2 66560611 IC50 = 0.95 nM T99041 C02XCY 66560612 IC50 = 0.56 nM T99041 CW64RD 66561555 IC50 > 100000 nM T99041 C9GTI7 66561556 IC50 > 100000 nM T99041 CC85DI 66561873 IC50 = 2.3 nM T99041 C0QCA2 66561874 IC50 = 3.8 nM T99041 C5F6NR 66896083 Ki = 4 nM T99041 COIA16 66953432 IC50 = 645 nM T99041 C8CMU1 66953714 IC50 = 9 nM T99041 CUR3E1 66954220 IC50 = 1.6 nM T99041 CFW13I 66954232 IC50 = 100 nM T99041 CJY9L6 66962050 IC50 > 5000 nM T99041 CVOH80 66963065 IC50 = 290 nM T99041 CX7Z8R 67506840 IC50 = 4.5 nM T99041 C7Y1PN 67507142 IC50 = 4.3 nM T99041 CUIB42 67507176 IC50 = 0.2 nM T99041 CF92IB 67507913 IC50 = 0.26 nM T99041 C9SND1 68305755 IC50 > 100000 nM T99041 CP3E2X 68416066 IC50 = 0.3 nM T99041 CX34PR 68417107 IC50 = 0.94 nM T99041 CCS6K9 68417211 IC50 = 0.63 nM T99041 CUKP32 68417894 IC50 = 15 nM T99041 C54VZI 68417897 IC50 = 5 nM T99041 C69VWN 68418230 IC50 = 0.85 nM T99041 C6K0XY 68418986 IC50 = 3.4 nM T99041 C6U9SP 68419033 IC50 = 12 nM T99041 CFNU91 68419172 IC50 = 2.9 nM T99041 CZ7QX8 68419268 IC50 = 4 nM T99041 CEF87L 68419860 IC50 = 0.62 nM T99041 CH3Z7F 68658979 IC50 = 0.14 nM T99041 C31XFM 68828690 IC50 = 140 nM T99041 C7X2WD 68828739 IC50 = 100 nM T99041 C4C3BL 68828935 IC50 = 9.2 nM T99041 CR27HN 68829000 IC50 = 7.5 nM T99041 CVGE51 68829025 IC50 = 28 nM T99041 CU4K6C 68829197 IC50 = 55 nM T99041 CP1NA4 68829414 IC50 = 4.6 nM T99041 C45ICV 68829529 IC50 = 250 nM T99041 C06ZLV 68829605 IC50 = 720 nM T99041 C2K3PM 68829714 IC50 = 13 nM T99041 CZOG14 68829854 IC50 = 510 nM T99041 C6R7ZV 68829908 IC50 = 540 nM T99041 C5I4BK 68829917 IC50 = 620 nM T99041 CCE26Z 68830038 IC50 = 52 nM T99041 C1HR3S 68830304 IC50 = 17 nM T99041 C47PHV 68830457 IC50 = 170 nM T99041 CYV1A0 68830878 IC50 = 6.8 nM T99041 C62LNY 68830888 IC50 = 0.38 nM T99041 CL1VS3 68832119 IC50 = 630 nM T99041 C6HRX1 68845950 IC50 = 56 nM T99041 CDJI62 68914093 IC50 = 8.2 nM T99041 C2TOQ7 69089363 IC50 = 60000 nM T99041 CO95AZ 69442708 IC50 = 23 nM T99041 CY98ML 69445181 IC50 = 1.1 nM T99041 C6BR4W 69445419 IC50 = 30 nM T99041 CD42CX 69446073 IC50 = 29 nM T99041 CS85UC 69446132 IC50 = 470 nM T99041 CZ49VQ 69446166 IC50 = 3.7 nM T99041 CFL92T 69446285 IC50 = 80 nM T99041 CXM07R 69446326 IC50 = 87 nM T99041 CWTN63 69446993 IC50 = 17 nM T99041 CBQJ90 69447448 IC50 = 19 nM T99041 C67CPF 69576646 IC50 = 45.3 nM T99041 CW4O2C 69689410 Ki = 34 nM T99041 CQ2DM1 69890803 Ki = 910 nM T99041 C0C8JW 70293564 IC50 = 200 nM T99041 CK26FY 70295607 IC50 = 4 nM T99041 CV4X5S 70295927 IC50 = 7 nM T99041 CXSV41 70296244 IC50 = 3 nM T99041 C3SB1V 70296823 IC50 = 40 nM T99041 CL64SQ 70297489 IC50 = 19900 nM T99041 CXD5V6 70297609 IC50 = 2 nM T99041 CEG1L5 70330884 IC50 = 23 nM T99041 C5W6LY 70681316 IC50 = 14 nM T99041 CLO96S 70681357 IC50 > 100000 nM T99041 CWP41T 70681469 IC50 > 100000 nM T99041 C7Z2KY 70681470 IC50 > 100000 nM T99041 C97JFS 70682267 IC50 = 17 nM T99041 CE1FU2 70682268 IC50 = 17 nM T99041 CI8EQ5 70682492 IC50 = 45.3 nM T99041 C03SDB 70682493 IC50 = 67.7 nM T99041 CF0U3A 70682494 IC50 = 57.6 nM T99041 C8Z2UQ 70682495 IC50 = 57.4 nM T99041 C14AWU 70682667 IC50 = 31 nM T99041 C71BSM 70682668 IC50 = 723 nM T99041 C49RIG 70682669 IC50 = 14.3 nM T99041 C19XIQ 70683454 IC50 > 100000 nM T99041 C07ADL 70683455 IC50 > 100000 nM T99041 C4YW5T 70684349 IC50 = 200 nM T99041 C6W1CT 70684350 IC50 = 18000 nM T99041 C1GF3E 70684351 IC50 = 53 nM T99041 C2GUS0 70684568 IC50 = 212 nM T99041 CU1I5S 70684569 IC50 = 39 nM T99041 CM96VS 70684570 IC50 = 47.7 nM T99041 C1NHS4 70684571 IC50 = 42.2 nM T99041 C7HF3B 70684748 IC50 = 298 nM T99041 C74WUS 70684749 IC50 = 879 nM T99041 CL8OZ4 70684750 IC50 = 10.3 nM T99041 CV5T8O 70684751 IC50 = 13.2 nM T99041 CO2NK6 70685557 IC50 > 100000 nM T99041 CK0WX8 70685558 IC50 > 100000 nM T99041 CLF84U 70685559 IC50 > 100000 nM T99041 C0K7PS 70685560 IC50 > 100000 nM T99041 C2T0NS 70685696 IC50 > 100000 nM T99041 C1Q3ZO 70686506 IC50 = 6.2 nM T99041 CM90BQ 70686720 IC50 = 264 nM T99041 CNQ50W 70686721 IC50 = 569 nM T99041 CRA4G1 70686722 IC50 = 64.6 nM T99041 C5I9BL 70686723 IC50 = 24.9 nM T99041 CT2LK4 70686905 IC50 = 104 nM T99041 CVD76F 70687705 IC50 > 100000 nM T99041 C28GVW 70687706 IC50 > 100000 nM T99041 CLQC52 70688610 IC50 = 29 nM T99041 C6MZ4N 70688809 IC50 = 101 nM T99041 C3GY6A 70688810 IC50 = 103 nM T99041 CGQV87 70688811 IC50 = 31.2 nM T99041 CHL1T9 70688964 IC50 = 320 nM T99041 C76SEY 70688965 IC50 = 28 nM T99041 CDVF75 70688966 IC50 = 715 nM T99041 CK2UC9 70688967 IC50 = 869 nM T99041 CI0VF5 70688968 IC50 = 843 nM T99041 C8K4WF 70688969 IC50 = 74 nM T99041 CVYH31 70689717 IC50 = 23 nM T99041 CUY81P 70689750 IC50 > 100000 nM T99041 CX2O0Z 70689751 IC50 > 100000 nM T99041 C17YKW 70689752 IC50 > 100000 nM T99041 CYO5X6 70690674 IC50 = 59 nM T99041 C2J7FS 70690675 IC50 = 15 nM T99041 CL6KR9 70690676 IC50 = 0.3 nM T99041 CXE41O 70690893 IC50 = 30.5 nM T99041 C4QCP6 70691068 IC50 = 863 nM T99041 C7ROY0 70691069 IC50 = 100 nM T99041 CC0D7S 70691070 IC50 = 34 nM T99041 C87LMG 70691901 IC50 > 100000 nM T99041 CL5EG7 70691902 IC50 > 100000 nM T99041 CGND49 70691903 IC50 > 100000 nM T99041 CGT57B 70691904 IC50 > 100000 nM T99041 CT89CW 70691905 IC50 > 100000 nM T99041 C5WI6V 70691906 IC50 > 100000 nM T99041 C19FJC 70692822 IC50 = 48 nM T99041 C8JZ3Q 70692823 IC50 = 16 nM T99041 C7FIR6 70693034 IC50 = 85.7 nM T99041 CM3L1E 70693035 IC50 = 50.4 nM T99041 C3DV6C 70693036 IC50 = 56.4 nM T99041 C3MF7C 70693037 IC50 = 91.5 nM T99041 C5YQ9B 70693038 IC50 = 33.9 nM T99041 CEQ4N8 70693039 IC50 = 76.2 nM T99041 CYQO06 70693040 IC50 = 36.7 nM T99041 C0S9LO 70693199 IC50 = 890 nM T99041 CY7M8K 70693200 IC50 = 19 nM T99041 C4P5TC 70693201 IC50 = 863 nM T99041 CEB6L2 70693202 IC50 = 116 nM T99041 CQMV53 70693949 IC50 > 100000 nM T99041 CBP8U7 70693950 IC50 > 100000 nM T99041 C0I2CV 70693951 IC50 > 100000 nM T99041 CCB64G 70693952 IC50 > 100000 nM T99041 C3ZUK2 70693953 IC50 > 100000 nM T99041 CS76EN 70693954 IC50 > 100000 nM T99041 C27PFC 70693955 IC50 > 100000 nM T99041 CVY48R 70693956 IC50 > 100000 nM T99041 CIX3F9 70694853 IC50 = 6.5 nM T99041 CQJD92 70694854 IC50 = 20 nM T99041 C8JRC5 70695073 IC50 = 99.7 nM T99041 CA0W8R 70695074 IC50 = 65.4 nM T99041 CYB1P3 70695075 IC50 = 74.4 nM T99041 C4ETL9 70695076 IC50 = 113.9 nM T99041 C5ZN7P 70695277 IC50 = 107 nM T99041 C3S5EX 70695278 IC50 = 26 nM T99041 CC6B7L 70695279 IC50 = 694 nM T99041 CXG5O4 70695280 IC50 = 311 nM T99041 CA01KO 70696068 IC50 > 100000 nM T99041 CSW43K 70696069 IC50 = 13100 nM T99041 C1NGL5 70696903 IC50 = 2.1 nM T99041 CR6FY8 70697121 IC50 = 194 nM T99041 C2B5UF 70697122 IC50 = 291 nM T99041 CV38GW 70697123 IC50 = 52.6 nM T99041 CJ4M0N 70697124 IC50 = 50.6 nM T99041 C4GIH1 70697292 IC50 = 31 nM T99041 CALB67 70697293 IC50 = 11.6 nM T99041 C19ZWC 70789754 IC50 > 100000 nM T99041 C31UTS 71184301 IC50 = 250 nM T99041 C8LY1U 71184352 IC50 = 9 nM T99041 C9IRW7 71184590 IC50 = 40 nM T99041 C8BK4O 71184607 IC50 = 4200 nM T99041 CS29MW 71184623 IC50 = 15700 nM T99041 C08NDK 71184749 IC50 = 20 nM T99041 CP91OE 71203742 IC50 = 625 nM T99041 CP6G5W 71203746 IC50 = 11.2 nM T99041 C32UMV 71203748 IC50 = 1.7 nM T99041 C04XQY 71203752 IC50 = 27.4 nM T99041 CE2I0K 71203758 IC50 = 123 nM T99041 CIQ7O2 71203767 IC50 = 13.5 nM T99041 C5GEJ9 71203769 IC50 = 156.1 nM T99041 C7LKV0 71203783 IC50 = 10.6 nM T99041 CBK26E 71449262 IC50 = 160 nM T99041 CW8JE0 71449264 IC50 = 150 nM T99041 CD9C3R 71449266 IC50 = 6900 nM T99041 CBX46U 71449270 IC50 = 54 nM T99041 CT35BK 71449272 IC50 = 64 nM T99041 C6D0WY 71449276 IC50 = 22 nM T99041 C46QSR 71449278 IC50 = 660 nM T99041 CKR1E6 71449280 IC50 = 72 nM T99041 CAJ8F0 71449608 IC50 = 20 nM T99041 CM5DB6 71450086 IC50 > 100000 nM T99041 CQU0Z1 71450087 IC50 > 100000 nM T99041 C65BCE 71450089 IC50 > 100000 nM T99041 CP9K2W 71450603 IC50 = 12 nM T99041 C8GBF1 71450604 IC50 = 670 nM T99041 CA3LP4 71450605 IC50 = 94 nM T99041 CD80JE 71451064 IC50 = 90 nM T99041 CH83NV 71451066 IC50 = 13 nM T99041 CM86TF 71451071 IC50 = 400 nM T99041 C9BK1J 71451073 IC50 = 17 nM T99041 CLC2N8 71451900 IC50 > 100000 nM T99041 CMU63C 71451901 IC50 > 100000 nM T99041 CT5WU4 71451902 IC50 > 100000 nM T99041 CL0X3F 71451939 IC50 > 100000 nM T99041 C7ZN6W 71452445 IC50 = 41 nM T99041 CKVA72 71452446 IC50 = 250 nM T99041 CP5NS6 71452447 IC50 = 110 nM T99041 C61LNR 71452448 IC50 = 83 nM T99041 C2J3GF 71452890 IC50 > 10000 nM T99041 C4GQ5B 71452892 IC50 = 90 nM T99041 CEM2O9 71453723 IC50 > 100000 nM T99041 CB1EX7 71453762 IC50 > 100000 nM T99041 CN4FE7 71454208 IC50 = 24 nM T99041 CD4IE2 71454659 IC50 = 3500 nM T99041 C2GO8L 71454668 IC50 = 12 nM T99041 CT9YS3 71454883 IC50 = 16 nM T99041 CBOK64 71455456 IC50 > 100000 nM T99041 CD32GT 71455458 IC50 > 100000 nM T99041 CQA9L7 71455494 IC50 > 100000 nM T99041 C1LRH5 71455960 IC50 = 84 nM T99041 CGH7R6 71455961 IC50 = 55 nM T99041 CGKJ82 71456385 IC50 = 38 nM T99041 CCY8P7 71456387 IC50 = 8900 nM T99041 CIC59O 71456389 IC50 = 3.8 nM T99041 CNGO29 71456391 IC50 = 60 nM T99041 C7AU4I 71456393 IC50 = 17 nM T99041 CVIF92 71456398 IC50 > 10000 nM T99041 C0CHQ9 71456400 IC50 = 66 nM T99041 C4T7CO 71457236 IC50 > 100000 nM T99041 C3GAO1 71457237 IC50 > 100000 nM T99041 CE3MP2 71457238 IC50 > 100000 nM T99041 C42BSO 71457239 IC50 > 100000 nM T99041 C8VI9L 71457240 IC50 > 50000 nM T99041 CK0O9D 71457760 IC50 = 490 nM T99041 C59TGZ 71457761 IC50 = 16 nM T99041 C8O6HJ 71457762 IC50 = 59 nM T99041 CBKA19 71457763 IC50 = 190 nM T99041 CI15BH 71457764 IC50 = 160 nM T99041 C5T6QP 71457765 IC50 = 72 nM T99041 C87VPZ 71458224 IC50 = 51 nM T99041 C89DPI 71458226 IC50 = 10 nM T99041 CK6S7X 71458227 IC50 = 6.3 nM T99041 CB67AV 71458229 IC50 = 3.5 nM T99041 CLRE92 71458241 IC50 = 66 nM T99041 CW76HL 71458243 IC50 = 16 nM T99041 CIO50T 71459090 IC50 > 100000 nM T99041 CXIM97 71459091 IC50 > 100000 nM T99041 CJ6N1C 71459092 IC50 > 100000 nM T99041 CUB4V8 71459679 IC50 = 7.8 nM T99041 C10JPO 71459680 IC50 = 330 nM T99041 CWQ59G 71460084 IC50 = 25 nM T99041 CZ7E1K 71460086 IC50 = 56 nM T99041 CS89OV 71460088 IC50 = 21 nM T99041 C6Z8RT 71460094 IC50 = 271 nM T99041 CKXG80 71460143 IC50 = 0.32 nM T99041 CEY13Z 71460148 IC50 = 6.3 nM T99041 CEU0B1 71460149 IC50 > 1000 nM T99041 CSC3I7 71460901 IC50 > 100000 nM T99041 CG7VX2 71460902 IC50 > 100000 nM T99041 C5K3WJ 71460903 IC50 > 100000 nM T99041 C3UF9P 71460904 IC50 > 100000 nM T99041 CUJT52 71461398 IC50 = 1100 nM T99041 CQ6GA0 71461399 IC50 = 50 nM T99041 CJ07GY 71461805 IC50 = 110 nM T99041 C8LB7A 71461808 IC50 = 11 nM T99041 C79EIW 71461811 IC50 = 1.6 nM T99041 CPAN79 71461821 IC50 = 3400 nM T99041 C02ALK 71461822 IC50 = 340 nM T99041 C7TS9F 71462596 IC50 > 100000 nM T99041 C63SUR 71462597 IC50 > 100000 nM T99041 CZT3S0 71462641 IC50 > 100000 nM T99041 CY2W5V 71463119 IC50 = 390 nM T99041 C16PTB 71463120 IC50 = 280 nM T99041 CKZ17B 71463121 IC50 = 60 nM T99041 C4VKM3 71463122 IC50 = 100 nM T99041 CY4W8D 71520057 IC50 = 660 nM T99041 C0JUM4 71520123 IC50 = 1320 nM T99041 CZ0UG8 71520163 IC50 = 720 nM T99041 CQO90M 71550930 IC50 = 1.55 nM T99041 C57JVN 71566829 Ki = 4 nM T99041 CMX9E3 71566830 Ki = 18 nM T99041 CDJ2T7 71566831 Ki = 14 nM T99041 C2SB3J 71566832 Ki = 18 nM T99041 C3J4DA 71566833 Ki = 11 nM T99041 CGVS23 71566834 Ki = 18 nM T99041 C5EQ8X 71566966 Ki = 13 nM T99041 C1VG2P 71566967 Ki = 30 nM T99041 C8FH4K 71566968 Ki = 8 nM T99041 C6AQ8P 71566969 Ki = 5 nM T99041 CM3NB6 71566970 Ki = 4 nM T99041 C92TKQ 71566971 Ki = 2 nM T99041 CZN30Q 71567105 Ki = 35 nM T99041 CL0BY5 71567106 Ki = 38 nM T99041 C63UAJ 71567107 Ki = 15 nM T99041 CPLH40 71567235 Ki = 10 nM T99041 CNM83T 71568676 Ki = 98 nM T99041 CEGB81 71568801 Ki = 75 nM T99041 C1G5WV 71568802 Ki = 25 nM T99041 CGXB93 71568803 Ki = 23 nM T99041 C0XK9O 71568804 Ki = 18 nM T99041 CL57TN 71568805 Ki = 14 nM T99041 CGJQ86 71568806 Ki = 18 nM T99041 CY3ZG6 71582959 IC50 = 211.9 nM T99041 C97MES 71583061 IC50 = 44 nM T99041 CB1YX0 71583062 IC50 = 44.1 nM T99041 CX43IU 71583063 IC50 = 27.6 nM T99041 C3KW9P 71583064 IC50 = 48.2 nM T99041 CEK26O 71583065 IC50 = 7.05 nM T99041 C53UMG 71583066 IC50 = 139.2 nM T99041 C9IRB0 71583175 IC50 = 60.1 nM T99041 CY87XJ 71583176 IC50 = 14.5 nM T99041 CD5O8F 71583177 IC50 = 52.6 nM T99041 C85BGF 71583178 IC50 = 11.4 nM T99041 CA67NL 71583179 IC50 = 4.67 nM T99041 C17-APR 71583292 IC50 = 5.93 nM T99041 CUH48W 71583293 IC50 = 15.5 nM T99041 C9AKS7 71594483 IC50 = 22390 nM T99041 C7B8AO 71621488 IC50 > 100000 nM T99041 C8T2PW 71655265 IC50 = 2800 nM T99041 CVB75Q 71655394 IC50 = 1800 nM T99041 CH4ZS0 71655395 IC50 > 100000 nM T99041 CC93KJ 71655554 IC50 > 100000 nM T99041 CN90KH 71655555 IC50 > 100000 nM T99041 CUT37D 71655556 IC50 > 100000 nM T99041 C71OFQ 71655557 IC50 > 100000 nM T99041 C7R6HU 71655622 IC50 > 100000 nM T99041 C2NA1M 71655623 IC50 > 100000 nM T99041 CDF08H 71655624 IC50 > 100000 nM T99041 CBEX27 71655625 IC50 > 100000 nM T99041 CT6XB5 71655626 IC50 > 100000 nM T99041 C1ND2P 71655627 IC50 > 100000 nM T99041 CXZ8N4 71667081 IC50 > 100000 nM T99041 CJ9QU7 71667226 IC50 > 100000 nM T99041 CE0Z8G 71667227 IC50 > 100000 nM T99041 CL7CS3 71667230 IC50 > 100000 nM T99041 CB6SI5 71667231 IC50 > 100000 nM T99041 C75UWV 71667375 IC50 > 100000 nM T99041 C19CTI 71667376 IC50 > 100000 nM T99041 C69CJB 71667378 IC50 > 100000 nM T99041 C07HNK 71667379 IC50 > 100000 nM T99041 CK74SP 71667380 IC50 > 100000 nM T99041 CMYZ68 71667381 IC50 > 100000 nM T99041 CDI39U 71667510 IC50 > 100000 nM T99041 CT49CO 71674688 IC50 = 34650 nM T99041 C8YTW3 71716406 Ki = 109 nM T99041 CQR5A1 71718946 IC50 = 460 nM T99041 CXKP89 71719452 Ki = 695 nM T99041 C0V3ZW 71720156 IC50 = 860 nM T99041 C0SC3Q 71720681 Ki = 1201 nM T99041 C7BD2R 71720854 IC50 = 2 nM T99041 CW3JG7 71731241 IC50 > 10000 nM T99041 C3D4HJ 71731243 IC50 = 31.3 nM T99041 CU6BC5 71731355 IC50 = 22 nM T99041 C5TS9Y 71731356 IC50 = 3.1 nM T99041 C5RTY9 71731357 IC50 = 3.4 nM T99041 CD9F5X 71731476 IC50 = 10.8 nM T99041 C3IO9H 71731477 IC50 = 6.6 nM T99041 CVAD62 71731478 IC50 = 2 nM T99041 C1ON0X 71731479 IC50 = 9.1 nM T99041 CZYQ05 71731604 IC50 = 1.9 nM T99041 C40YRO 71731605 IC50 = 0.7 nM T99041 C9Q8MO 72164809 IC50 = 9.39 nM T99041 CL5X1Z 72164811 IC50 = 25.5 nM T99041 C7N8WB 72164813 IC50 = 17.61 nM T99041 C2R0NV 72164815 IC50 = 8.28 nM T99041 C4JLM5 72164817 IC50 = 19.54 nM T99041 C6RQ9A 72164819 IC50 = 7.56 nM T99041 C38GWP 72164942 IC50 = 3.79 nM T99041 C4T0MY 72164944 IC50 = 15.24 nM T99041 C0T4UW 72164946 IC50 = 10.45 nM T99041 CLV02R 72164948 IC50 = 6.05 nM T99041 CHPN10 72164950 IC50 = 20.84 nM T99041 CI78FQ 72165082 IC50 = 7.5 nM T99041 CN0VU2 72165084 IC50 = 4.35 nM T99041 C84SYX 72165086 IC50 = 8.57 nM T99041 C1RQA3 72165088 IC50 = 10.02 nM T99041 CH51ZR 72165090 IC50 = 15.7 nM T99041 C1HL2A 72188903 IC50 = 13100 nM T99041 CLS1A0 72188904 IC50 > 100000 nM T99041 CO15AV 72188905 IC50 = 0.66 nM T99041 CPDC28 72188906 IC50 = 140 nM T99041 CL7P3D 72193502 IC50 = 24400 nM T99041 C4AXB8 72193503 IC50 = 38000 nM T99041 CQC28P 72193504 IC50 = 2800 nM T99041 CV87PE 72193505 IC50 = 26600 nM T99041 C65DFP 72697059 IC50 = 18 nM T99041 CX07OC 72697060 IC50 = 248 nM T99041 CZ56DO 72697061 IC50 = 11 nM T99041 C1A2KX 72697062 IC50 = 17 nM T99041 CS5U1F 72697063 IC50 = 29 nM T99041 CA3HI1 72697064 IC50 = 75 nM T99041 CCZJ47 72697206 IC50 = 20 nM T99041 CWNZ91 72697207 IC50 = 21 nM T99041 C6BWI4 72697208 IC50 = 31 nM T99041 C9JA1Q 72697209 IC50 = 4 nM T99041 CF6A8N 72697210 IC50 = 4 nM T99041 CTMR03 72697211 IC50 = 42 nM T99041 CP9NV5 72697212 IC50 = 27 nM T99041 C1P8HS 72697352 IC50 = 46 nM T99041 CC7G3M 72697353 IC50 = 63 nM T99041 CXYO73 72697354 IC50 = 209 nM T99041 CAXV78 72697355 IC50 = 17 nM T99041 CGV09W 72697356 IC50 = 3 nM T99041 CIF9D7 72697357 IC50 = 4 nM T99041 CC8RA6 72697358 IC50 = 15 nM T99041 C1EC7S 72697359 IC50 = 292 nM T99041 C8CRO6 72697494 IC50 = 5 nM T99041 C03NKY 72697495 IC50 = 6 nM T99041 CP0MU3 72697496 IC50 = 125 nM T99041 CI60AK 72697497 IC50 = 94 nM T99041 CO19YK 72697498 IC50 = 22 nM T99041 C47IGZ 72697499 IC50 = 20 nM T99041 C65OPG 72697500 IC50 = 6 nM T99041 C3ZP7N 72697501 IC50 = 23 nM T99041 C7EF8C 72697646 IC50 = 60 nM T99041 C08IGP 72699737 IC50 = 1.98 nM T99041 CMT61I 72707535 IC50 = 198 nM T99041 CAEF04 72707536 IC50 = 2177.5 nM T99041 C7ARW4 72707537 IC50 = 1.2 nM T99041 C8D5PB 72725804 IC50 = 11900 nM T99041 CC10AZ 73345857 IC50 > 100000 nM T99041 CSZR98 73346173 IC50 = 48 nM T99041 C1L4RX 73346174 IC50 = 1 nM T99041 CX4F0Y 73347359 IC50 > 100000 nM T99041 C3XFM5 73347360 IC50 > 100000 nM T99041 CGNL10 73347698 IC50 = 720 nM T99041 CR09PJ 73348871 IC50 > 10000 nM T99041 CA79DR 73349143 IC50 = 265 nM T99041 CO5TB8 73349220 IC50 = 37 nM T99041 C06WRM 73350448 IC50 > 100000 nM T99041 C1T7LK 73350449 IC50 > 100000 nM T99041 CCIZ12 73350450 IC50 > 100000 nM T99041 CNC6B8 73350798 IC50 = 125 nM T99041 CDBV29 73350799 IC50 = 27 nM T99041 CYG04J 73352283 IC50 = 12600 nM T99041 CFV5U3 73353424 IC50 > 100000 nM T99041 CRS4O0 73353425 IC50 > 100000 nM T99041 C7X9ZG 73353601 IC50 > 1000 nM T99041 CV6BA3 73353756 IC50 = 37 nM T99041 C51QGP 73353757 IC50 = 27 nM T99041 CBK37N 73353758 IC50 = 64 nM T99041 CLYP23 73354936 IC50 > 100000 nM T99041 CLO76J 73355285 IC50 = 11 nM T99041 CCVT96 73355286 IC50 = 1.6 nM T99041 CH9W2R 73356494 IC50 > 100000 nM T99041 CKD46T 73356495 IC50 > 100000 nM T99041 CI0N6E 73356496 IC50 > 10000 nM T99041 C7R3ZT 76309823 Ki = 142000 nM T99041 CY0N9K 76311138 IC50 = 170 nM T99041 CWK7M6 76311139 IC50 = 50 nM T99041 CF5S9X 76313540 Ki = 61000 nM T99041 CIP4R0 76314754 IC50 = 40 nM T99041 C3HRA1 76314755 IC50 = 50 nM T99041 C1ZAC3 76317994 IC50 = 113760 nM T99041 C68JOX 76318341 IC50 = 30 nM T99041 CET31O 76318342 Ki = 3.5 nM T99041 CP0H8I 76320760 Ki = 4500 nM T99041 C9UGA3 76325642 IC50 = 113600 nM T99041 CNIP02 76325643 IC50 = 5 nM T99041 C08DYM 76325644 IC50 = 120 nM T99041 C3C7HE 76325645 Ki = 9 nM T99041 CWBL62 76327979 Ki = 6300 nM T99041 CW4M6E 76329221 IC50 = 390 nM T99041 C3LPR2 76331631 Ki = 5000 nM T99041 C7S6EY 76332265 IC50 = 4364 nM T99041 CH95ZJ 76336484 IC50 = 520 nM T99041 C4W7RE 77461184 IC50 = 8.5 nM T99041 CRG30N 86267497 IC50 = 148 nM T99041 C7JRH1 86267498 IC50 = 89.6 nM T99041 CTXI04 86267501 IC50 = 3 nM T99041 CO78UK 86267502 IC50 = 3.4 nM T99041 C7K2NA 86267708 IC50 = 3.8 nM T99041 CPS4U2 86268135 IC50 = 2290 nM T99041 C9GA1T 86268138 IC50 = 299 nM T99041 CBJ6N8 86268336 IC50 = 19.2 nM T99041 CA3L2Q 86268337 IC50 = 15.4 nM T99041 C6HCF9 86268525 IC50 = 18.6 nM T99041 CLG83C 86268944 IC50 = 4.9 nM T99041 C31OGJ 86279928 IC50 = 10.8 nM T99041 CB60OP 89488720 IC50 = 2.6 nM T99041 CIV7Y8 89668929 IC50 > 100000 nM T99041 C87GJT 89704940 IC50 > 100000 nM T99041 CHI7U9 89704942 IC50 > 100000 nM T99041 CSLI09 89704955 IC50 > 100000 nM T99041 CA3K7R 89704970 IC50 > 100000 nM T99041 CF89OD 89705045 IC50 > 100000 nM T99041 CK3Z8J 89705076 IC50 > 100000 nM T99041 CH6P0S 89705081 IC50 > 100000 nM T99041 C63DGS 89705096 IC50 > 100000 nM T99041 CND56S 89705098 IC50 > 100000 nM T99041 C0CKQ7 89705100 IC50 > 100000 nM T99041 C0CPD1 89705103 IC50 > 100000 nM T99041 C1IL7N 89705109 IC50 > 50000 nM T99041 CA48MR 89705136 IC50 > 100000 nM T99041 C5F9OA 89705152 IC50 > 100000 nM T99041 C1VSG5 89705179 IC50 > 100000 nM T99041 CHAS49 89705195 IC50 > 100000 nM T99041 C0RP1J 89705223 IC50 > 100000 nM T99041 CQO0I6 89705242 IC50 > 100000 nM T99041 C7DF1P 89705244 IC50 > 100000 nM T99041 C03OGJ 89705273 IC50 > 100000 nM T99041 CGX4I7 89705275 IC50 = 19000 nM T99041 CX9BC3 89712515 IC50 > 100000 nM T99041 CM5N8H 90654714 IC50 = 1436 nM T99041 CFY63H 90654715 IC50 = 378 nM T99041 CC6VX3 90654716 IC50 = 382 nM T99041 CA0SL5 90654717 IC50 = 342 nM T99041 CAM68Q 90654718 IC50 = 217 nM T99041 CQ93MA 90654719 IC50 = 193 nM T99041 CNDG24 90654720 IC50 = 1388 nM T99041 CC46WF 90654721 IC50 = 452 nM T99041 CCX20I 90654722 IC50 = 443 nM T99041 COV32D 90654723 IC50 = 404 nM T99041 CZ7KU8 90654724 IC50 = 885 nM T99041 CUH0W7 90654725 IC50 = 910 nM T99041 CCX14G 90654726 IC50 = 1034 nM T99041 CXUY06 90654727 IC50 = 1023 nM T99041 CKC94W 90654728 IC50 = 997 nM T99041 C8VBP2 90654729 IC50 = 119 nM T99041 C2UN8K 90654730 IC50 = 84 nM T99041 C1GSQ3 90654731 IC50 = 77.6 nM T99041 C47YVG 90654732 IC50 = 122 nM T99041 C20CDE 90654733 IC50 = 79 nM T99041 C9B2MJ 90654734 IC50 = 74 nM T99041 C30OWT 90654735 IC50 = 157 nM T99041 C3XP8C 90654736 IC50 = 119 nM T99041 CQD53I 90654737 IC50 = 125 nM T99041 C10TVX 90654738 IC50 = 111 nM T99041 C17RCY 90654739 IC50 = 19 nM T99041 CLT2X9 90654740 IC50 = 197 nM T99041 CDO0J4 90654741 IC50 = 148 nM T99041 CS62OC 90654742 IC50 = 134 nM T99041 C4B8KC 90654743 IC50 = 137 nM T99041 CKU5M8 90654744 IC50 = 43 nM T99041 C6TGZ5 90655538 IC50 > 100000 nM T99041 C9P3HJ 90655539 IC50 > 100000 nM T99041 CT98OM 90655540 IC50 > 100000 nM T99041 CVQ8M4 90655541 IC50 > 100000 nM T99041 CT6Q2L 90655542 IC50 > 100000 nM T99041 C7Z4GV 90655543 IC50 > 100000 nM T99041 CE3HC2 90655544 IC50 > 100000 nM T99041 CU2I3V 90655545 IC50 > 100000 nM T99041 C2NZ7X 90655546 IC50 > 100000 nM T99041 C0E5UP 90655547 IC50 > 100000 nM T99041 CF23RI 90655548 IC50 > 100000 nM T99041 CW3QG7 90655549 IC50 > 100000 nM T99041 CHG4E2 90655550 IC50 > 100000 nM T99041 CTA78W 90655551 IC50 > 100000 nM T99041 CA6S4W 90655552 IC50 > 100000 nM T99041 C3LT0S 90655553 IC50 > 100000 nM T99041 CEW45X 90655554 IC50 > 100000 nM T99041 CRX52D 90655555 IC50 > 100000 nM T99041 C9KG1U 90655556 IC50 > 100000 nM T99041 CXYE76 90655557 IC50 > 100000 nM T99041 CES85Q 90655558 IC50 > 100000 nM T99041 CK7IB9 90655559 IC50 >= 100000 nM T99041 CAG5X4 90655560 IC50 > 100000 nM T99041 C3IJA0 90655561 IC50 > 100000 nM T99041 C4V0ZY 90655562 IC50 > 100000 nM T99041 CY9G8Q 90655563 IC50 > 100000 nM T99041 CPIN84 90664318 IC50 = 53 nM T99041 CY76CR 90664436 IC50 = 1.8 nM T99041 C8YPL7 90664437 IC50 = 11 nM T99041 CU9LB2 90664438 IC50 > 100000 nM T99041 CQ20XA 90664578 IC50 > 100000 nM T99041 CV87ZH 90664579 IC50 > 100000 nM T99041 C9OC4Q 90664688 IC50 = 8.1 nM T99041 CJVF52 90664689 IC50 = 19 nM T99041 CDEN13 90664693 IC50 > 100000 nM T99041 CFG21I 90664805 IC50 = 2.9 nM T99041 C37YWE 90664828 IC50 = 84 nM T99041 CP60NA 90664941 IC50 = 7.8 nM T99041 CJ04US 90664942 IC50 = 69 nM T99041 CCH31U 90665060 IC50 = 23 nM T99041 C4LB2V 90665061 IC50 = 17 nM T99041 C0C1VT 90665186 IC50 = 12 nM T99041 CJ81VK 90665187 IC50 = 73 nM T99041 CHB2D6 90666864 IC50 = 16580 nM T99041 CFH71J 91937923 IC50 = 3730 nM T99041 COA7Z6 92131131 IC50 = 14 nM T99041 CBQ38C 101879512 IC50 = 170 nM T99041 CM7E4V 101887269 IC50 > 50000 nM T99041 C8EH0J 101887270 IC50 = 5.8 nM T99041 CDT67J 101887271 IC50 = 25 nM T99041 C4F2CS 101887272 IC50 > 100000 nM T99041 C58XWA 101887273 IC50 = 18100 nM T99041 C3Y9ET 101887274 IC50 > 100000 nM T99041 C1AF8C 101887275 IC50 = 1440 nM T99041 CH7QC5 101887276 IC50 > 50000 nM T99041 CO4FR2 101887277 IC50 = 29 nM T99041 C9JEH0 101887278 IC50 = 13900 nM T99041 C52GIO 101887279 IC50 > 100000 nM T99041 CO95EZ 118705501 IC50 = 570 nM T99041 CH8VO2 118705502 IC50 = 30 nM T99041 CZ1G3O 118712516 IC50 > 100000 nM T99041 C8X4JA 118712517 IC50 > 100000 nM T99041 CC29AB 118712518 IC50 > 100000 nM T99041 CB09PD 118712519 IC50 > 100000 nM T99041 CD4U1X 118712520 IC50 > 100000 nM T99041 CU0V5J 118712521 IC50 > 100000 nM T99041 C03OUP 118712522 IC50 > 100000 nM T99041 CT2MZ8 118712764 IC50 = 450 nM T99041 C3W5RU 118712765 IC50 = 220 nM T99041 CKA1N5 118712766 IC50 = 160 nM T99041 C8M6ZW 118712767 IC50 = 220 nM T99041 CV5C6D 118712768 IC50 = 320 nM T99041 C2NSC7 118712769 IC50 = 430 nM T99041 CV8JY3 118712770 IC50 = 640 nM T99041 C4KCZ1 118712771 IC50 = 770 nM T99041 CAR4W5 118712772 IC50 = 40 nM T99041 CRWT85 118712773 IC50 = 530 nM T99041 C36YUB 118712774 IC50 = 1580 nM T99041 C4T2FY 118712775 IC50 = 50 nM T99041 C0MYA1 118712776 IC50 = 1940 nM T99041 C8IF4E 118712777 IC50 = 440 nM T99041 CJ8EL0 118712778 IC50 = 70 nM T99041 C07UOL 118712779 IC50 = 360 nM T99041 C25HYG 118712780 IC50 = 130 nM T99041 CD0HQ4 118712781 IC50 = 270 nM T99041 C5D9RH 118712782 IC50 = 8800 nM T99041 CB7NX6 118712783 IC50 = 1980 nM T99041 C46TMQ 118712785 IC50 = 70 nM T99041 CA1I4M 118712786 IC50 = 47440 nM T99041 CUN79Q 118712787 IC50 = 9650 nM T99041 C5M3BX 118712788 IC50 = 10 nM T99041 CV3AK9 118717414 IC50 = 2390 nM T99041 C1NAQ9 118717415 IC50 > 100000 nM T99041 CKES65 118717416 IC50 > 100000 nM T99041 CYP07B 118719171 Ki = 6000 nM T99041 CD3L8W 118719172 Ki = 520 nM T99041 C8WJL2 118719173 Ki = 900 nM T99041 C5HU8M 118719174 Ki = 2700 nM T99041 C36XYR 118722404 IC50 = 5810 nM T99041 CX6J2E 118722405 IC50 = 340 nM T99041 C7BD8K 118722406 IC50 = 380 nM T99041 C0K6YG 118722407 IC50 = 760 nM T99041 CK7HN4 118722408 IC50 = 70 nM T99041 CFV6N4 118722409 IC50 = 3660 nM T99041 CK71WT 118722410 IC50 = 70 nM T99041 CI74ZM 118722411 IC50 = 80 nM T99041 CH1P7Y 118722412 IC50 = 70 nM T99041 CL8TY5 118722413 IC50 = 180 nM T99041 CGK98I 118722414 IC50 = 320 nM T99041 CBK91L 118722415 IC50 = 510 nM T99041 C8KUP0 118722416 IC50 = 290 nM T99041 C76DBO 118722417 IC50 = 540 nM T99041 CW6L5X 118722418 IC50 = 330 nM T99041 CM6Y5I 118722419 IC50 = 430 nM T99041 C37BGF 118722420 IC50 = 610 nM T99041 COG4V6 118722421 IC50 = 140 nM T99041 CIQ5Z7 118722422 IC50 = 430 nM T99041 CH6GX2 118728164 IC50 = 6 nM T99041 CFCI13 118728166 IC50 = 4.7 nM T99041 CS08AG 118728168 IC50 = 1.4 nM T99041 C0AG2Q 118728920 IC50 = 500 nM T99041 CE1ZS2 118728922 IC50 = 230 nM T99041 CVG84E 118728927 IC50 = 640 nM T99041 CBI68Y 118728931 IC50 = 36 nM T99041 CI0E1U 118736611 IC50 = 695 nM T99041 C2NX7C 118736612 IC50 = 2801 nM T99041 CP71VU 118736613 IC50 = 27.54 nM T99041 CL40TU 118736614 IC50 = 145 nM T99041 CJI2B8 118736615 IC50 = 85 nM T99041 C15XMK 118736616 IC50 = 108 nM T99041 C1IGJ6 118736617 IC50 = 67 nM T99041 C4BI2T 118736618 IC50 = 258 nM T99041 CED50R 118736620 IC50 = 100 nM T99041 C3DT9O 118736622 IC50 = 94 nM T99041 C6TYS7 122172854 IC50 = 4376 nM T99041 C2U5PE 122178432 IC50 = 20 nM T99041 C7TEY3 122178433 IC50 = 19.8 nM T99041 C8OLP9 122178434 IC50 = 346 nM T99041 C9GP3L 122178435 IC50 = 2.9 nM T99041 C8P2DB 122178436 IC50 = 6.4 nM T99041 CGFU89 122178437 IC50 = 3.4 nM T99041 CN78TQ 122189864 IC50 = 650 nM T99041 CNM82F 122189865 IC50 > 100000 nM T99041 C19GHJ 122189866 IC50 = 12200 nM T99041 C3U9KC 122189867 IC50 > 100000 nM T99041 CW5V3U 122189868 IC50 = 180 nM T99041 CCG05R 122189869 IC50 = 1800 nM T99041 CI01PT 122189870 IC50 = 180 nM T99041 C80EWF 122189871 IC50 = 220 nM T99041 C3N7JC 122189872 IC50 > 100000 nM T99041 CG8O1J 122189873 IC50 > 100000 nM T99041 CK0US2 122189874 IC50 = 980 nM T99041 C5V6NI 122189875 IC50 > 100000 nM T99041 CV7A9Y 122189876 IC50 > 100000 nM T99041 CN86VR 122189878 IC50 > 100000 nM T99041 C24OVE 122190735 IC50 = 1320 nM T99041 CSN6E0 122190738 IC50 = 24000 nM T99041 CD4EF9 122190739 IC50 = 1060 nM T99041 CVU5G7 122190835 IC50 = 2230 nM T99041 CB5X2Q 122190838 IC50 = 100000 nM T99041 CG69FQ 122190841 IC50 = 1250 nM T99041 CJ7X2U 122194794 IC50 = 1.5 nM T99041 C8XVB4 122194795 IC50 = 290 nM T99041 CL43TO 122194796 IC50 = 0.8 nM T99041 CAPX63 126456388 IC50 = 2.06 nM T99041 C0DUI4 126842756 IC50 = 1.33 nM T99041 CZXV13 126842761 IC50 = 0.76 nM T99041 CF7KI9 126842762 IC50 = 1.62 nM T99041 CG93JS 126842771 IC50 = 1.22 nM T99041 C6PLX9 127035081 IC50 = 4.9 nM T99041 CJ0KS7 127035239 IC50 = 2.3 nM T99041 CKSZ13 127035240 IC50 = 1.8 nM T99041 C6T1IM 127035241 IC50 = 5.7 nM T99041 CJRL72 127035242 IC50 = 0.7 nM T99041 CVKI59 127035243 IC50 = 1.9 nM T99041 CWJX95 127035244 IC50 = 2.3 nM T99041 C0XMS7 127035375 IC50 = 1.9 nM T99041 CMK5Q9 127035376 IC50 = 1.4 nM T99041 C4N7QB 127035377 IC50 = 1.6 nM T99041 CGN49F 127035378 IC50 = 4.3 nM T99041 C36UHW 127035569 IC50 = 0.3 nM T99041 CTKS36 127035740 IC50 = 3.7 nM T99041 CAXT02 127035741 IC50 = 3.2 nM T99041 CZB0L6 127035742 IC50 = 1.1 nM T99041 C4QWL5 127035743 IC50 = 1.3 nM T99041 CPGF39 127035744 IC50 = 1.8 nM T99041 CXTD34 127035745 IC50 = 1.8 nM T99041 CM98XR 127035752 IC50 = 1.7 nM T99041 C87MVA 127035753 IC50 = 1.7 nM T99041 CDW25O 127035754 IC50 = 0.4 nM T99041 CN08IS 127045827 IC50 > 100000 nM T99041 CAK85G 127046590 IC50 > 50000 nM T99041 CP3U8J 127046622 IC50 > 100000 nM T99041 CFAI71 127046624 IC50 = 56000 nM T99041 CB6PA7 127046626 IC50 > 100000 nM T99041 C76IGF 127046628 IC50 > 100000 nM T99041 CHL49F 127046630 IC50 = 790 nM T99041 CH0D2Z 127046632 IC50 = 4000 nM T99041 CK4SO7 127047730 IC50 = 2600 nM T99041 CSO9L3 127047731 IC50 = 19400 nM T99041 C4KIA9 127047732 IC50 = 16200 nM T99041 CHX41E 127047733 IC50 = 680 nM T99041 C6I7HW 127047734 IC50 = 34000 nM T99041 C2CP4F 127047761 IC50 > 100000 nM T99041 CYR1X2 127047762 IC50 > 100000 nM T99041 CIV4C2 127047839 IC50 > 100000 nM T99041 CDYA70 127047985 IC50 > 100000 nM T99041 C0FS5E 127048116 IC50 > 100000 nM T99041 C6NIM5 127048874 IC50 = 8.6 nM T99041 CXD69M 127048875 IC50 = 289 nM T99041 C65MAC 127048876 IC50 = 44 nM T99041 C23BWQ 127049179 IC50 = 1.4 nM T99041 CNCB06 127049180 IC50 = 1.9 nM T99041 CJ8SG3 127049204 IC50 = 1.5 nM T99041 CRM04V 127049507 IC50 = 0.5 nM T99041 C76VPA 127049823 IC50 = 54 nM T99041 CH0X6Q 127050132 IC50 = 0.5 nM T99041 CIGA32 127050759 IC50 = 1.1 nM T99041 CNY90B 127050760 IC50 = 1.5 nM T99041 C80WCY 127050761 IC50 = 0.6 nM T99041 CUVQ34 127050762 IC50 = 2.9 nM T99041 CJMS57 127051032 IC50 = 1.1 nM T99041 C9V4EG 127051045 IC50 = 0.7 nM T99041 C7W8JR 127051639 IC50 = 699 nM T99041 C36SXH 127052286 IC50 = 1.1 nM T99041 CBR1F8 127052287 IC50 = 26 nM T99041 CHZX75 127052288 IC50 = 0.6 nM T99041 CB34GQ 127052289 IC50 = 0.7 nM T99041 CLG0Q3 127052290 IC50 = 16 nM T99041 CL2S0F 127052581 IC50 = 1.7 nM T99041 C1W5AL 127052582 IC50 = 155 nM T99041 C4TI8H 127052590 IC50 = 1170 nM T99041 CNV0A8 127052636 IC50 = 0.56 nM T99041 CS2Z9R 127052637 IC50 = 0.23 nM T99041 C75EAL 127052638 IC50 = 0.24 nM T99041 CRP1K2 130385241 IC50 = 5.8 nM T99041 CTIO26 130385242 IC50 = 5.17 nM T99041 C30ERZ 130385243 IC50 = 1.9 nM T99041 C09MJL 130385246 IC50 = 205.2 nM T99041 CZ29WO 130385251 IC50 = 19.64 nM T99041 CED01R 130385253 IC50 = 14.95 nM T99041 C83CDX 130385258 IC50 = 8.42 nM T99041 CB37AX 130385267 IC50 = 216.2 nM T99041 C5DWM6 130391940 IC50 = 70.42 nM T99041 C41QVU 130391961 IC50 = 6.13 nM T99041 C6PMX7 130391978 IC50 = 17.65 nM T99041 CD7B2H 130392003 IC50 = 8.91 nM T99041 C15BEV 130392042 IC50 = 563.9 nM T99041 CD6C4U 130392043 IC50 = 13070 nM T99041 CH9E4W 132055397 IC50 = 110.1 nM T99041 C6CV5J 132069286 IC50 = 154.67 nM T99041 CALB73 134131859 IC50 = 5400 nM T99041 CA5Y0V 134132454 IC50 = 250 nM T99041 CMY0V5 134132485 IC50 = 5000 nM T99041 CTZU69 134132901 IC50 = 14.6 nM T99041 CH1G3A 134133219 IC50 = 260 nM T99041 CS9K7A 134133834 IC50 = 360 nM T99041 C2BA5L 134134276 IC50 = 890 nM T99041 CVE96U 134134571 IC50 = 300 nM T99041 CB59UX 134135207 IC50 = 73 nM T99041 CIXJ53 134135875 IC50 = 250 nM T99041 C4Q2GB 134136466 IC50 = 121.56 nM T99041 C5OS4T 134136634 IC50 = 39.2 nM T99041 C14XET 134137196 IC50 = 140 nM T99041 CMB8T7 134137851 IC50 = 32.64 nM T99041 CTP9X4 134138048 IC50 = 21520 nM T99041 C58KIQ 134138807 IC50 = 500 nM T99041 C2OWQ1 134138838 IC50 = 760 nM T99041 CPLI26 134139792 IC50 = 400 nM T99041 CDV6U9 134140856 IC50 = 49.73 nM T99041 C5TS2J 134141415 IC50 = 2600 nM T99041 CB8QD9 134142015 IC50 = 770 nM T99041 CY2CJ4 134142362 IC50 = 510 nM T99041 CK27IY 134143858 IC50 = 2930 nM T99041 CKP0Z5 134144315 IC50 = 78.33 nM T99041 COT7P4 134144691 IC50 = 206.71 nM T99041 CD0XT6 134145610 IC50 = 800 nM T99041 C8B3CU 134150931 IC50 = 280 nM T99041 CEC9Y2 134151020 IC50 = 50860 nM T99041 C0G5PV 134151859 IC50 = 220 nM T99041 C3NF8J 134151937 IC50 = 140 nM T99041 CQRM94 134152842 IC50 = 360 nM T99041 C6TL9Z 134153173 IC50 = 950 nM T99041 CBN6Z7 134153444 IC50 = 610 nM T99041 CZX9V0 134154214 IC50 = 337.8 nM T99041 C4ZWS1 134157002 IC50 = 120 nM T99041 CNO0R1 135411740 IC50 = 2120 nM T99041 CRM4Q8 135518358 IC50 = 3 nM T99041 CMI5A6 135964368 IC50 = 95 nM T99041 CC4L2F 136060652 IC50 > 3000 nM T99041 CP7BS2 136098501 IC50 = 6113 nM T99041 CO04QA 136177302 IC50 = 7 nM T99041 C1GYM8 136411530 IC50 = 11 nM T99041 CR4VI2 137225025 IC50 = 0.6 nM T99041 CAN18C 137631813 IC50 = 2.1 nM T99041 C95BML 137632265 IC50 = 70 nM T99041 C5H2EA 137637131 IC50 = 27.54 nM T99041 C2FA1T 137637208 IC50 = 7.2 nM T99041 CS2L6B 137637588 IC50 = 43.4 nM T99041 CO9BH6 137638100 IC50 = 50.2 nM T99041 C6IJ3A 137642352 IC50 = 8.5 nM T99041 CY0R4C 137644720 IC50 = 60 nM T99041 CI8FG2 137644837 IC50 = 1200 nM T99041 C1MBC4 137646578 IC50 = 31.8 nM T99041 C67NZA 137650009 IC50 = 123.3 nM T99041 C8BH1R 137650030 IC50 = 537 nM T99041 CG8HS3 137652269 IC50 = 29 nM T99041 C9SX0Q 137653253 IC50 = 139 nM T99041 CH4MT1 137655300 IC50 = 8.7 nM T99041 CV5A3F 137657117 IC50 = 470 nM T99041 CKF03W 137659671 IC50 = 5.5 nM T99041 C2MV9K 137661375 IC50 = 151.7 nM T99041 CJT56Y 137662038 IC50 = 2.6 nM T99041 CO6JA3 141514759 IC50 = 188.7 nM T99041 C1SQ2R 141514762 IC50 = 64.47 nM T99041 CHI84B 141514764 IC50 = 65.36 nM T99041 C3SKH4 145948172 IC50 = 97 nM T99041 C8S7FY 145949528 IC50 = 1.45 nM T99041 CR2UP9 145950777 IC50 > 100 nM T99041 C7IZU2 145950786 IC50 = 1.61 nM T99041 C7SMW4 145951086 IC50 = 0.72 nM T99041 CR5AJ7 145952072 IC50 = 26.6 nM T99041 C2MWR4 145952134 IC50 = 15.3 nM T99041 CV30OD 145952476 IC50 = 0.77 nM T99041 CBFR49 145953292 IC50 = 1.69 nM T99041 CYF24S 145953544 IC50 = 0.76 nM T99041 C38IOE 145953726 IC50 = 0.61 nM T99041 C4JQT5 145953757 IC50 > 100 nM T99041 C0C4KJ 145954860 IC50 = 0.79 nM T99041 C48AXH 145955793 IC50 = 2.4 nM T99041 C6QY1K 145957483 IC50 = 1.58 nM T99041 CMO0J1 145957949 IC50 = 1.67 nM T99041 C35FNU 145957994 IC50 = 18 nM T99041 CR9S6F 145958227 IC50 = 2.3 nM T99041 CB72HG 145958828 IC50 = 1.25 nM T99041 C60WXK 145959997 IC50 = 0.77 nM T99041 C8V5PA 145962482 IC50 = 0.54 nM T99041 CBL76R 145964231 IC50 = 2500 nM T99041 CF53NA 145964407 IC50 = 400 nM T99041 CNMT16 145965136 IC50 = 1200 nM T99041 CQW63D 145965301 IC50 = 11500 nM T99041 C6D0VY 145967130 IC50 = 21500 nM T99041 CI82EJ 145973071 IC50 = 10400 nM T99041 C1Y5FP 145973406 IC50 = 6.8 nM T99041 CP8EN1 145973616 IC50 = 0.54 nM T99041 CP7VT2 145973710 IC50 = 1300 nM T99041 C2C1ZR 145974002 IC50 = 17200 nM T99041 C9C4WU 145975568 IC50 = 80 nM T99041 CRNK53 145977284 IC50 = 46500 nM T99041 CWF4Y7 145977953 IC50 = 2000 nM T99041 CB3K0Q 145978529 IC50 = 59900 nM T99041 CR3I9D 145978547 IC50 = 49 nM T99041 CNG4Z2 145983347 IC50 = 1.12 nM T99041 CH6P8Q 145983352 IC50 = 1270 nM T99041 C02BLT 145983464 IC50 = 7580 nM T99041 CN1V6D 145984069 IC50 = 28050 nM T99041 C3QT0G 145984247 IC50 = 1780 nM T99041 CMWH26 145984429 IC50 = 15780 nM T99041 CL6D3F 145984547 IC50 = 19.6 nM T99041 CIX4P5 145985997 IC50 = 232.8 nM T99041 CM6L4K 155510749 IC50 = 190 nM T99041 C5ZQ7W 155511281 IC50 = 2.91 nM T99041 CP4SH8 155511399 IC50 > 100000 nM T99041 CEL39X 155511987 IC50 = 74.6 nM T99041 CQA73O 155512586 IC50 = 197 nM T99041 C57QZJ 155512836 IC50 = 7.6 nM T99041 CX3U8Z 155515016 IC50 = 10.21 nM T99041 C7FOS5 155516136 IC50 = 538 nM T99041 CTE94M 155516800 IC50 > 10000 nM T99041 C19ZCJ 155518265 IC50 = 395 nM T99041 C8UOJ4 155518381 IC50 = 1.7 nM T99041 C8U9ON 155518908 Ki = 217.9 nM T99041 CW0NI8 155519444 IC50 = 0.1 nM T99041 C7O2UF 155519988 IC50 > 100000 nM T99041 C3I8AW 155520161 IC50 = 60 nM T99041 C1Z2NP 155522069 Ki = 152.8 nM T99041 C4AZ9V 155523785 IC50 = 93.2 nM T99041 CG18KV 155524302 IC50 = 0.75 nM T99041 C0RAC6 155524362 IC50 = 3900 nM T99041 CTSA30 155526359 IC50 = 5.61 nM T99041 CVD89H 155526728 IC50 = 208 nM T99041 C5C4UV 155526759 IC50 = 5.99 nM T99041 CAT3J0 155526949 IC50 = 3.9 nM T99041 C7J4VQ 155527859 IC50 = 1.75 nM T99041 CLE9I0 155528648 IC50 = 0.22 nM T99041 C3LT9C 155529752 IC50 > 100000 nM T99041 C8FHJ2 155529886 IC50 = 2.43 nM T99041 CCX9H6 155530472 IC50 = 226 nM T99041 C7YP3B 155530585 IC50 = 4.41 nM T99041 C2YWG1 155530817 IC50 = 790 nM T99041 CB6N4S 155531120 IC50 = 0.18 nM T99041 CGV6C1 155531169 IC50 = 22.09 nM T99041 CEOQ32 155531330 IC50 = 50.9 nM T99041 CMY59I 155531892 IC50 > 100000 nM T99041 C0ZCE3 155533243 IC50 = 89.8 nM T99041 CN04KW 155533304 IC50 = 74.43 nM T99041 C95ZUT 155534726 Ki = 180.8 nM T99041 CW8Z1X 155535213 IC50 > 100000 nM T99041 CA9Z6Q 155538747 IC50 = 121300 nM T99041 CG3RS6 155540249 IC50 = 223 nM T99041 CJ67GL 155540375 IC50 = 3.5 nM T99041 CM1FA9 155544265 Ki = 380.1 nM T99041 CY25EZ 155544299 IC50 = 4.6 nM T99041 C8H3MJ 155544665 IC50 = 20.48 nM T99041 CU17DA 155544967 IC50 = 2.35 nM T99041 CY2V6P 155545256 IC50 = 2.25 nM T99041 C62YMT 155545522 IC50 = 85.48 nM T99041 CMS63L 155545906 IC50 = 56.6 nM T99041 CGZ08R 155547532 IC50 = 3830000 nM T99041 CDGW26 155547608 IC50 = 76170 nM T99041 CNA9X4 155548276 IC50 = 217 nM T99041 CWF0L6 155548277 IC50 = 483 nM T99041 CM9K4B 155548792 IC50 = 0.72 nM T99041 CB1AF4 155549522 IC50 = 7.5 nM T99041 CL9R1Y 155549582 IC50 > 100000 nM T99041 C3MW1B 155550953 IC50 > 10000 nM T99041 CX9Y4B 155552378 IC50 = 1.05 nM T99041 C8XSI3 155553379 IC50 = 2 nM T99041 C6QKL9 155553392 Ki = 412.2 nM T99041 C1D5QZ 155554658 IC50 = 2.5 nM T99041 CR8AU9 155555628 IC50 = 68510 nM T99041 C1GD0E 155555672 Ki = 941.2 nM T99041 CHV85S 155556058 IC50 > 100000 nM T99041 C6N4WH 155557237 IC50 > 100000 nM T99041 CSCD34 155559193 IC50 > 100000 nM T99041 C7KVR5 155559306 IC50 = 3.9 nM T99041 CRL47X 155559391 IC50 = 28.7 nM T99041 C1NE4T 155560255 IC50 > 100000 nM T99041 C68CRH 155561682 IC50 = 4 nM T99041 CQ7JL5 155562412 IC50 = 55870 nM T99041 C90QLF 155563643 Ki = 103.7 nM T99041 C48ETF 155565121 IC50 = 170 nM T99041 CUL27B 155565517 Ki = 341.6 nM T99041 CE5SI7 155566076 IC50 > 100000 nM T99041 CI5C6P 155568161 IC50 = 0.44 nM T99041 CUQL05 155568269 IC50 = 5.06 nM T99041 CDB0S2 155568427 IC50 = 421 nM T99041 D00HSG 44408767 IC50 = 3300 nM T99041 D00KMP 44431763 IC50 = 5300 nM T99041 D00RIX 5280443 IC50 = 140 nM T99041 D00YEV 5281605 IC50 > 200000 nM T99041 D02RDY 11375559 IC50 > 100000 nM T99041 D02RIE 44440628 Ki = 13000 nM T99041 D02WBC 3847395 IC50 = 33000 nM T99041 D03DNV 71655266 IC50 > 100000 nM T99041 D04CAR 10607286 Ki = 0.4 nM T99041 D05LYC 11403745 IC50 = 140 nM T99041 D05UUA 16049437 Ki = 820 nM T99041 D05XWX 10130510 Ki = 3.8 nM T99041 D06AUB 44440618 Ki = 3400 nM T99041 D06NRU 1393052 IC50 = 2300 nM T99041 D06UKY 44440632 Ki = 2800 nM T99041 D07ALM 11232124 Ki = 0.082 nM T99041 D07HWI 6931234 IC50 = 75000 nM T99041 D07IJU 13578534 Ki = 2100 nM T99041 D08NMS 46900258 Ki = 1.4 nM T99041 D09ALJ 5280805 IC50 = 145000 nM T99041 D09BYA 44431745 IC50 = 3500 nM T99041 D09MVE 263366 IC50 = 30000 nM T99041 D0AU0M 637542 IC50 = 83180 nM T99041 D0CP1J 56658139 IC50 > 50000 nM T99041 D0G3TK 5280863 IC50 = 132000 nM T99041 D0JI3S 11674875 IC50 = 18600 nM T99041 D0JL2T 5393152 IC50 > 200000 nM T99041 D0L5RI 44328273 Ki = 7880 nM T99041 D0L9XR 447256 Ki = 470 nM T99041 D0N1FU 6918465 Ki = 126 nM T99041 D0N1QQ 94701 Ki = 2200 nM T99041 D0N5CI 11615508 IC50 = 12000 nM T99041 D0O9RD 44403067 Ki = 3350 nM T99041 D0P5OE 2724998 IC50 = 45000 nM T99041 D0PB2M 23645372 Ki = 34 nM T99041 D0R5OE 44422449 IC50 = 538 nM T99041 D0S0RK 10680 IC50 = 170 nM T99041 D0T2EW 11075394 Ki = 1.4 nM T99041 D0T3PW 5281672 IC50 = 37150 nM T99041 D0U4HG 23634523 IC50 > 36900 nM T99041 D0V9EN 689043 IC50 = 3370 nM T99041 D0W4GM 205131 IC50 = 40000 nM T99041 D0X0IF 23655936 IC50 > 39100 nM T99041 D0X2JG 2777206 IC50 = 37000 nM T99041 D0Y3TZ 370 IC50 = 4650 nM T99041 D0Y5IQ 44255320 IC50 = 10000 nM T28043 D05PZB 135398495 IC50 = 1 nM T28043 D0E3TC 44259 IC50 = 0.227 nM T28043 D03BNU 59604787 IC50 > 10000 nM T28043 C3I5CX 304956 IC50 = 860 nM T28043 CK9P4E 348062 IC50 = 590 nM T28043 CC5NB0 348063 IC50 = 470 nM T28043 CUT16A 594733 IC50 = 4300 nM T28043 CW75MC 687283 IC50 = 520 nM T28043 C0YXB7 709463 IC50 = 2830 nM T28043 C2JAQ8 723792 IC50 = 4310 nM T28043 CLUR08 739692 IC50 = 8740 nM T28043 COA87I 2731384 IC50 = 790 nM T28043 CACS26 11561968 Ki > 2000 nM T28043 CU0E8O 11690457 Ki = 940 nM T28043 CB0AP2 11705863 Ki > 2000 nM T28043 C5IHO2 24800600 IC50 = 20 nM T28043 C1NKE3 46905987 IC50 = 850 nM T28043 C1MR8Q 60097495 IC50 > 10000 nM T28043 CV63UL 67240318 IC50 > 10000 nM T28043 CY8BZ9 72771105 IC50 = 20 nM T28043 CG16YE 72771106 IC50 = 4 nM T28043 C23OUG 90645197 IC50 = 10 nM T28043 C53PWG 90645198 IC50 = 40 nM T28043 C01WEM 90645199 IC50 = 40 nM T28043 C5K7RU 90645200 IC50 = 50 nM T28043 CG9TO6 90645201 IC50 = 70 nM T28043 C95HNS 90645202 IC50 = 210 nM T28043 C03WJT 90645203 IC50 = 220 nM T28043 C42BKF 90645204 IC50 = 220 nM T28043 CK30AI 90645205 IC50 = 340 nM T28043 C1D6NT 90645206 IC50 = 410 nM T28043 C8H1JX 90645207 IC50 = 490 nM T28043 CYK2P3 90645208 IC50 = 560 nM T28043 CKQ40O 90645209 IC50 = 620 nM T28043 C49ZDO 90645210 IC50 = 620 nM T28043 CN8L4E 90645211 IC50 = 730 nM T28043 C18DTQ 90645212 IC50 = 970 nM T28043 C1SHE5 90645213 IC50 = 1000 nM T28043 C58CQS 90645214 IC50 = 1100 nM T28043 C2E6UD 90645215 IC50 = 1200 nM T28043 C38OTD 90645216 IC50 = 1400 nM T28043 C2IHG1 90645217 IC50 = 2800 nM T28043 CBG09A 90645218 IC50 = 3200 nM T28043 CYK85Z 90645219 IC50 = 4000 nM T28043 CM0K2F 90645220 IC50 = 9300 nM T28043 C9W5LQ 127029823 IC50 = 15 nM T28043 CR6MO9 127030141 IC50 = 2160 nM T28043 C67TOM 127030142 IC50 = 1340 nM T28043 CQ6Z5M 127030143 IC50 = 4580 nM T28043 CPU0O5 127030414 IC50 = 590 nM T28043 C4CXH7 127030458 IC50 = 1010 nM T28043 C2LN0P 127034074 IC50 = 3530 nM T28043 CT2K3V 127034326 IC50 = 3500 nM T28043 CC95UA 127034332 IC50 = 990 nM T28043 C2MD1Q 155513187 IC50 > 10000 nM T28043 D09PTP 57325421 IC50 = 7 nM T28043 D0M5FF 5083 IC50 = 10 nM T58307 CKA6I1 5703330 IC50 = 10800 nM T58307 C62ZXE 44607965 IC50 = 600 nM T58307 D0YH7K 24856225 IC50 = 10 nM T20761 CUXI92 70681359 IC50 = 0.32 nM T20761 CW8N5L 71042827 IC50 = 0.3 nM T20761 CX9Q5J 90057788 IC50 = 0.47 nM T20761 C7T9FK 90654562 IC50 = 0.12 nM T06455 D00YZD 54726191 IC50 > 100000 nM T06455 D05BMG 3007 IC50 = 3500 nM T06455 D06HLY 5910 Ki = 3000 nM T06455 D08SKH 4114 Ki = 250 nM T06455 D09XQF 3767 Ki = 60000 nM T06455 D0K9MY 11243969 IC50 > 50000 nM T06455 D0T8GD 89594 Ki = 4400 nM T06455 D0TY5N 854019 IC50 = 35000000 nM T06455 D0Y3KG 3121 Ki = 9150000 nM T06455 D00VUI 6199 Ki = 600 nM T06455 D06ZEO 54674461 IC50 > 50000 nM T06455 D07AOL 16741 Ki = 1700 nM T06455 D08CJK 1150 Ki = 1700 nM T06455 D08VSQ 59336911 IC50 > 40000 nM T06455 D0M9RQ 11697697 IC50 > 27000 nM T06455 D0QR5G 2355 Ki = 12000 nM T06455 D0V9VG 51049968 IC50 >= 20000 nM T06455 D09SWE 31244 IC50 = 5150 nM T06455 D0D3GL 137662068 IC50 > 40000 nM T06455 D0LU9X 74221950 IC50 > 50000 nM T06455 D04RLX 148201 IC50 > 100000 nM T06455 D06ZVC 10150497 IC50 = 41000 nM T06455 C4N9ZB 240 IC50 = 3920 nM T06455 C5WI3K 408 IC50 = 34994516.7 nM T06455 C2H5PB 931 IC50 = 25003.45 nM T06455 C93REJ 995 IC50 = 97000 nM T06455 C4DS3F 2361 IC50 > 25000 nM T06455 C9OY1P 4685 IC50 = 16982.44 nM T06455 C3LCS1 7002 IC50 = 33962.53 nM T06455 C7J3QE 7003 IC50 = 17988.71 nM T06455 CK1GM9 7005 IC50 = 130000 nM T06455 C01EVA 7055 IC50 = 2398.83 nM T06455 CZU01G 7056 IC50 = 5395.11 nM T06455 CKGX24 7060 IC50 = 190000 nM T06455 CC9UD1 7119 IC50 = 62000 nM T06455 C9C6AL 7138 IC50 = 400000 nM T06455 CA8DB1 7479 Ki = 3600 nM T06455 CG98SM 7724 IC50 = 8100 nM T06455 C9GPQ1 7725 IC50 = 4880 nM T06455 C95TVD 7804 IC50 = 59000 nM T06455 CK1F8C 8663 IC50 = 139958.73 nM T06455 CD6IX9 10249 Ki = 7500 nM T06455 CEA89F 10256 Ki = 11000 nM T06455 C8H4SX 10724 IC50 = 51999.6 nM T06455 C8ZQX7 11306 IC50 = 30974.19 nM T06455 C9KBP8 11317 IC50 = 26000 nM T06455 C0R1KU 11326 IC50 = 31000 nM T06455 C1G2AL 11327 IC50 = 8298.51 nM T06455 C8T9PF 11328 IC50 = 130016.96 nM T06455 CLY6K9 11372 IC50 = 549.54 nM T06455 CVO8C2 11387 IC50 = 10000 nM T06455 C7IA9M 11389 Ki = 7700 nM T06455 C6S7NL 11396 IC50 = 1698.24 nM T06455 C29BVT 11926 IC50 = 199986.19 nM T06455 C6WES0 13414 IC50 = 279898.13 nM T06455 CTX63M 13652 IC50 = 11994.99 nM T06455 CVQ2U6 14306 IC50 = 25000 nM T06455 C5PE3W 14536 IC50 = 830000 nM T06455 C9VSI5 15592 IC50 = 60000 nM T06455 CD28UY 15768 IC50 = 2500 nM T06455 CJQ9W6 15769 IC50 = 2500.35 nM T06455 CK8VZ4 16309 IC50 = 14996.85 nM T06455 C43QPK 16312 IC50 > 60000 nM T06455 CF76BS 16323 IC50 = 149968.48 nM T06455 CK3OJ7 16619 IC50 > 100000 nM T06455 C42VKG 24905 IC50 = 6400 nM T06455 CYM2U8 38950 IC50 = 52000 nM T06455 CPT5G4 61341 IC50 = 17000 nM T06455 CW03PD 66042 IC50 > 100000 nM T06455 C65HZQ 67583 IC50 = 670 nM T06455 C0FK8W 68266 IC50 = 20989.4 nM T06455 C95JWC 68487 Ki = 1100 nM T06455 CO0HB3 75473 Ki = 3300 nM T06455 C6NUX9 76751 IC50 = 5300 nM T06455 CB7J3G 77409 Ki = 27000 nM T06455 C5VB1P 91393 IC50 = 7400 nM T06455 CC0P7F 94378 IC50 > 30000 nM T06455 CMA78T 95864 IC50 > 100000 nM T06455 CYIJ31 96389 IC50 = 1800 nM T06455 CMKQ41 114908 IC50 > 600000 nM T06455 CO31SB 139097 IC50 = 900 nM T06455 C3C0VD 151091 Ki = 64800 nM T06455 C9SEK0 157672 IC50 = 580000 nM T06455 CK8RD5 168114 IC50 = 59000 nM T06455 CJ34CF 168115 IC50 = 98300 nM T06455 CMA9N8 227328 IC50 = 1600 nM T06455 CV9U4J 237074 Ki = 10 nM T06455 CH37CT 249266 IC50 = 35974.93 nM T06455 C7YM0E 289925 Ki = 2400 nM T06455 C0LT3C 317317 IC50 = 88000 nM T06455 C1B9YV 329983 Ki = 840 nM T06455 CVFB56 442478 Ki = 2000 nM T06455 CD5HT1 589040 Ki = 70 nM T06455 C6R5XN 595145 Ki = 1200 nM T06455 CVRM18 595254 Ki = 220 nM T06455 CH81ZF 609844 IC50 = 1999861.87 nM T06455 C82CVS 659526 IC50 > 100000 nM T06455 C1M0CH 676494 IC50 > 100000 nM T06455 CF5QZ4 693141 IC50 = 500 nM T06455 C0NQO8 736499 IC50 > 100000 nM T06455 CGW2Y5 736500 Ki = 130 nM T06455 CZG18E 1201554 Ki = 4100 nM T06455 CKF67B 2733992 IC50 = 34000 nM T06455 CE94ON 2763178 Ki = 8600 nM T06455 C0AR8P 2773435 IC50 = 1500 nM T06455 CQ9NZ8 2773875 IC50 = 50 nM T06455 CJF32C 2776125 IC50 = 41000 nM T06455 CW1GX5 2776264 IC50 = 140000 nM T06455 CR1N5T 2776335 IC50 = 18000 nM T06455 C2YNT0 2776338 IC50 = 270000 nM T06455 C5IB1P 2776342 IC50 = 37000 nM T06455 CR5M0P 2776347 IC50 = 1500 nM T06455 CZF61B 2779861 IC50 = 51000 nM T06455 CST09R 2794770 IC50 = 3400 nM T06455 C0ZUR9 2794830 Ki = 3300 nM T06455 CRC56T 2795184 Ki = 100 nM T06455 CKR58B 2795448 IC50 = 600 nM T06455 C8IV9A 2795535 IC50 = 72000 nM T06455 CG2X7K 2795537 IC50 < 100000 nM T06455 C4A7TL 2795538 IC50 < 100000 nM T06455 C5IE0J 2798782 Ki = 90 nM T06455 CFC9M0 2806034 IC50 > 100000 nM T06455 CAJQ53 3040177 Ki = 250 nM T06455 CO18WM 4730695 Ki = 620 nM T06455 CZM7D8 5281794 IC50 = 83300 nM T06455 C48OIX 7074967 Ki = 12800 nM T06455 CR01AH 7537465 Ki = 800 nM T06455 C7I5CK 7537499 IC50 = 500 nM T06455 C54TBK 7537503 Ki = 200 nM T06455 COC24T 7537534 IC50 = 680 nM T06455 CA15IT 9796590 IC50 > 30000 nM T06455 CXD39F 10081254 Ki = 6300 nM T06455 C4A5SP 10379988 IC50 > 10000 nM T06455 C8TPU0 10510985 Ki = 890 nM T06455 CJPW17 10654534 Ki = 22700 nM T06455 CP25XG 10702138 IC50 = 11000 nM T06455 CX4HA8 10749527 Ki = 60 nM T06455 CZS9Q5 10899427 Ki = 790 nM T06455 C1A8HL 11171679 Ki = 14200 nM T06455 C9PT1B 11182787 Ki = 3200 nM T06455 C1XR3I 11206290 Ki = 20 nM T06455 C03XEJ 11206520 Ki >= 67000 nM T06455 CJ1O6V 11207072 Ki = 230 nM T06455 C3U5QZ 11217334 Ki >= 67000 nM T06455 CMHY80 11229234 Ki = 280 nM T06455 C7LK3C 11276492 Ki = 4500 nM T06455 CIUE57 11290471 Ki = 1500 nM T06455 CF5YS9 11310529 Ki = 22200 nM T06455 C60BAD 11311338 Ki = 1500 nM T06455 CMQD35 11321674 Ki = 180 nM T06455 CU72EY 11344157 Ki = 130 nM T06455 C5FG8X 11355925 IC50 = 4200 nM T06455 C1BOK3 11378800 Ki = 250 nM T06455 CZIC23 11389737 Ki = 970 nM T06455 CYL06Q 11389927 IC50 = 1300 nM T06455 CN0UM2 11446630 Ki = 35200 nM T06455 CW57BU 11480732 Ki = 520 nM T06455 CU3X5J 11701255 Ki = 44500 nM T06455 C54DUQ 11785088 Ki = 2800 nM T06455 C6A1LM 11786814 IC50 > 500000 nM T06455 C5HDW9 11816351 Ki = 5600 nM T06455 C1T8XZ 11993865 Ki = 400 nM T06455 CBZ83S 11993868 Ki = 6200 nM T06455 C7A1EZ 11993870 Ki = 300 nM T06455 C4XP2N 11993872 Ki = 800 nM T06455 CWT0S3 11993875 Ki = 600 nM T06455 C3E2PJ 12215260 Ki >= 67000 nM T06455 C0DG7E 13349626 Ki = 5100 nM T06455 CN52YX 13349629 Ki = 1800 nM T06455 C7I9PF 13557523 Ki = 6600 nM T06455 C7PMK9 14345241 Ki = 9800 nM T06455 CB26ML 14835679 IC50 = 8400 nM T06455 CM0VL2 15543761 Ki = 2700 nM T06455 C28ZJD 15563485 IC50 = 6700 nM T06455 CT4RL1 15778480 Ki = 1400 nM T06455 CUDC52 16037176 Ki = 43700 nM T06455 CJU50N 16072099 IC50 > 100000 nM T06455 C8D0KF 16099905 IC50 = 20000 nM T06455 C2FXW0 16099923 IC50 = 500000 nM T06455 C8FLH6 16202152 IC50 > 10000 nM T06455 CL0R4J 16244360 Ki = 1400 nM T06455 C76RIB 16654683 Ki = 27400 nM T06455 CVJ4O1 16654686 Ki = 250 nM T06455 CA3JQ1 16654687 Ki = 6200 nM T06455 C9C5TV 17751819 IC50 > 50000 nM T06455 COY3E2 18351319 IC50 < 100000 nM T06455 C48BGL 20440932 Ki = 70 nM T06455 CDL4G9 23645678 IC50 > 200000 nM T06455 CR9ZI2 24764491 IC50 > 50000 nM T06455 CF7ON5 25099235 IC50 > 50000 nM T06455 C27LVU 25817326 Ki = 19700 nM T06455 CS40ML 44123747 IC50 > 50000 nM T06455 C6FA8R 44388586 Ki = 9700 nM T06455 CC17PX 44388593 Ki = 6600 nM T06455 CM6V4C 44388606 Ki = 130 nM T06455 CKV1H9 44388612 Ki = 170 nM T06455 CGU79D 44388657 IC50 = 3700 nM T06455 CVU5K0 44388702 Ki = 11000 nM T06455 CTI5R6 44388718 Ki = 170 nM T06455 CAWL05 44428924 IC50 > 100000 nM T06455 CW9V1F 45117642 IC50 = 1500 nM T06455 CO3P0J 46866604 IC50 > 30000 nM T06455 CX18GT 46889932 IC50 > 10000 nM T06455 CF14PE 46947264 IC50 > 30000 nM T06455 CJD25G 52920263 IC50 = 16000 nM T06455 CUIB93 56679632 IC50 = 9800 nM T06455 CY58ZD 57330086 IC50 = 106000 nM T06455 C37SMZ 57505249 IC50 > 100000 nM T06455 C7I4QD 57519510 IC50 > 50000 nM T06455 C9ZE7J 58874273 IC50 > 50000 nM T06455 CTL97W 60151476 IC50 > 45000 nM T06455 CE18JH 60202715 Ki = 2180 nM T06455 CFM6H7 67049587 IC50 > 100000 nM T06455 C1EHX3 67306704 IC50 = 1000 nM T06455 C47GYB 71454279 IC50 > 10000 nM T06455 C4GNJ3 71598545 IC50 > 10000 nM T06455 CC07KL 71662263 IC50 > 25000 nM T06455 CO1B9W 71662264 IC50 > 25000 nM T06455 CI0VR5 71662265 IC50 > 25000 nM T06455 CHW2T7 71662266 IC50 > 25000 nM T06455 CY9VC3 71662267 IC50 > 25000 nM T06455 C1MHC9 71662268 IC50 > 25000 nM T06455 CO57BK 71662269 IC50 > 25000 nM T06455 CZ01TB 71662427 IC50 > 25000 nM T06455 CHKX52 71662428 IC50 > 25000 nM T06455 C6PF9B 71662429 IC50 > 25000 nM T06455 C3DZ1E 71662430 IC50 > 25000 nM T06455 CPH76Z 71662431 IC50 > 25000 nM T06455 CKQ42X 71662432 IC50 > 25000 nM T06455 CXFB14 71662433 IC50 > 25000 nM T06455 CJHI28 71770158 IC50 > 20000 nM T06455 C9LU5Q 71770282 IC50 > 20000 nM T06455 CWT7K2 72205601 IC50 > 20000 nM T06455 C3J0ZB 72725671 IC50 > 20000 nM T06455 C9WY3B 73386689 Ki = 710 nM T06455 CPG73S 73417116 Ki = 130 nM T06455 CZ3TB5 74221949 IC50 > 50000 nM T06455 CW9N8T 74222036 IC50 > 50000 nM T06455 CSDY49 82596666 IC50 = 5200 nM T06455 CN9MO7 86271494 IC50 >= 19000 nM T06455 CE4IT5 90408860 IC50 >= 19000 nM T06455 CB41MH 118560618 IC50 > 100000 nM T06455 CC6J8R 118722716 Ki = 500 nM T06455 CK3SI7 118722717 IC50 = 6600 nM T06455 C6TBD2 121345502 IC50 > 50000 nM T06455 C1C9LI 122246967 IC50 = 160 nM T06455 CUV9B7 127037739 Ki = 1.73 nM T06455 C4ONR3 127038432 Ki = 2.58 nM T06455 C8A2ZM 127038433 Ki = 3.07 nM T06455 C1QA7G 127038434 Ki = 6.02 nM T06455 CC1PB3 127038435 Ki = 2.7 nM T06455 CE4MN8 127038436 Ki = 13.2 nM T06455 C7QX5G 127038437 Ki = 3.27 nM T06455 CVH62U 127038438 Ki = 10.97 nM T06455 C8T1CN 127038439 Ki = 1.54 nM T06455 CZQ14B 127038440 Ki = 2.57 nM T06455 CD8FG2 127038811 Ki = 12.96 nM T06455 CCU5X6 127038814 Ki = 3.41 nM T06455 CKH20R 127038815 Ki = 0.057 nM T06455 CAG2L3 127038816 Ki = 16.62 nM T06455 CBP9S2 127042311 Ki = 1.93 nM T06455 CLT73G 137647199 IC50 > 10000 nM T06455 CXJ07F 145949470 IC50 = 550 nM T06455 CI3V6Y 145950358 IC50 = 55 nM T06455 CLZ54T 145950740 IC50 = 440 nM T06455 C4FM3C 145951105 IC50 = 830 nM T06455 CLV0G6 145951167 IC50 = 390 nM T06455 C3URG5 145951186 IC50 > 10000 nM T06455 CA9N2R 145951417 IC50 > 10000 nM T06455 CG5OW3 145951998 IC50 = 590 nM T06455 C4LJV9 145952024 IC50 = 330 nM T06455 C1QA6W 145952070 IC50 = 51 nM T06455 CC7IP8 145952109 IC50 = 670 nM T06455 C9D5MZ 145952745 IC50 = 3400 nM T06455 CRN85T 145952991 IC50 = 1300 nM T06455 CA7W2O 145953059 IC50 = 140 nM T06455 CCZ67T 145953474 IC50 > 10000 nM T06455 C5LB7M 145953999 IC50 = 380 nM T06455 CN5L4K 145954640 IC50 = 110 nM T06455 CQ5SN1 145955289 IC50 = 160 nM T06455 C7N6CA 145956935 IC50 = 76 nM T06455 C82NJA 145957007 IC50 > 10000 nM T06455 CBFU43 145957229 IC50 = 17 nM T06455 C20EDK 145957568 IC50 = 460 nM T06455 C3B0YE 145957778 IC50 = 560 nM T06455 CID3G5 145958087 IC50 = 5500 nM T06455 CZX8P9 145958165 IC50 > 10000 nM T06455 CM8U9A 145958674 IC50 = 290 nM T06455 CBF54O 145958967 IC50 = 1000 nM T06455 CB5XW7 145959080 IC50 = 400 nM T06455 CLS3W5 145959177 IC50 = 2700 nM T06455 CLJE41 145959897 IC50 = 3600 nM T06455 CW1GO5 145960043 IC50 = 130 nM T06455 CDKY72 145960338 IC50 = 1200 nM T06455 CZ83QK 145960490 IC50 > 50000 nM T06455 CKLA91 145962920 IC50 = 42 nM T06455 CXF9E7 145972420 IC50 = 410 nM T06455 C56HYE 145974067 IC50 = 220 nM T06455 CJN96Q 145974556 IC50 = 300 nM T06455 C9H1VK 155556442 IC50 > 50000 nM T06455 D01ARE 44388719 Ki = 590 nM T06455 D01UYI 5281607 IC50 > 25000 nM T06455 D02EAP 11993867 Ki = 13900 nM T06455 D06QFO 11332763 Ki = 40 nM T06455 D06TRS 23646069 Ki = 100 nM T06455 D0D5YP 5280371 Ki = 11600 nM T06455 D0I7GE 11790 IC50 > 25000 nM T06455 D0J1IE 11993873 Ki = 800 nM T06455 D0M0IQ 11210706 Ki = 1200 nM T06455 D0O1HH 11263510 Ki = 90 nM T06455 D0Q6PI 1001 IC50 = 4410 nM T06455 D0VD5O 11148236 Ki = 210 nM T06455 D0YP4A 11993866 Ki < 800 nM T06455 D0YQ8U 11993871 Ki = 600 nM T97917 C93RAZ 285404 EC50 = 170 nM T97917 C8FH4M 310357 EC50 = 4850 nM T97917 C1EC2Q 457933 EC50 = 1 nM T97917 CDO59A 708867 EC50 = 10000 nM T97917 CHTK06 727813 EC50 = 900 nM T97917 C8J0BH 735751 EC50 > 10000 nM T97917 CZ0VA4 872695 EC50 = 3000 nM T97917 CA16XZ 909951 EC50 = 1260 nM T97917 COB3P0 1098728 EC50 > 10000 nM T97917 CEF21T 1131797 EC50 = 6000 nM T97917 CSX6N0 1240119 EC50 = 90 nM T97917 CMG2I8 1292869 EC50 = 770 nM T97917 C59IPT 1367800 EC50 = 490 nM T97917 C62OTF 1416500 EC50 = 4030 nM T97917 CI2F3R 2054164 EC50 > 10000 nM T97917 CNY91H 2165902 EC50 = 3200 nM T97917 CYRS24 2211856 EC50 = 5880 nM T97917 CB70YI 2215592 EC50 = 3700 nM T97917 C3SVM7 2302157 EC50 = 4700 nM T97917 CC2NW4 4776370 EC50 = 8000 nM T97917 CO36UL 5308652 EC50 = 2730 nM T97917 C3J9CE 8005184 EC50 > 10000 nM T97917 CJ4Z6T 11418989 EC50 = 40 nM T97917 C0CUZ2 16036926 EC50 = 30 nM T97917 C4AT8U 16143873 IC50 = 60 nM T97917 CDSG62 22430370 EC50 = 100 nM T97917 CIK71E 22430372 EC50 = 12300 nM T97917 CXF3R5 22430395 EC50 = 980 nM T97917 CH2DI1 24776342 EC50 > 10000 nM T97917 CIAE78 24776344 EC50 = 5100 nM T97917 C13HPO 24776345 EC50 = 1020 nM T97917 CMN49A 24776346 EC50 = 690 nM T97917 C5GOM9 24776347 EC50 = 830 nM T97917 CKN8F9 24776348 EC50 = 1520 nM T97917 CKXA38 24776349 EC50 = 2710 nM T97917 CUK30M 24776350 EC50 = 130 nM T97917 C1H3PU 24776351 EC50 = 34 nM T97917 CV26ST 24776352 EC50 = 3500 nM T97917 CGH24A 24776353 EC50 = 1490 nM T97917 CMU90L 24776354 EC50 = 14100 nM T97917 CC5LJ6 24776355 EC50 = 810 nM T97917 C69CTS 24776356 EC50 = 12200 nM T97917 C5HVI6 24776357 EC50 = 270 nM T97917 C90PWR 24776358 EC50 = 1870 nM T97917 CKG2W3 25238441 EC50 = 100 nM T97917 C56OWF 44232675 EC50 = 4500 nM T97917 CJK72M 44232677 EC50 = 12300 nM T97917 CN74MP 44232924 EC50 = 5400 nM T97917 C2MP3Y 44232925 EC50 = 600 nM T97917 CAO83Q 44233644 EC50 = 1800 nM T97917 C3UBZ9 44233645 EC50 = 600 nM T97917 CJ6A2K 44233646 EC50 = 1100 nM T97917 CN81VH 44233647 EC50 = 1200 nM T97917 CMY4B3 44233648 EC50 = 1900 nM T97917 CXZ1K2 44233905 EC50 = 2400 nM T97917 C8S4IJ 44236326 EC50 = 2100 nM T97917 CP2R7H 44236328 EC50 = 1600 nM T97917 C8KW7R 44236329 EC50 = 8200 nM T97917 CCX6A4 44236330 EC50 = 900 nM T97917 CZ8D0C 44413496 EC50 = 250 nM T97917 CQ2B7I 44413497 EC50 = 80 nM T97917 CGD1U9 44413498 EC50 = 44 nM T97917 C6KF7I 44413499 EC50 = 1470 nM T97917 CX4EL0 44413507 EC50 = 540 nM T97917 CRI4V3 44413508 EC50 = 43 nM T97917 CV7K1U 44413524 EC50 = 140 nM T97917 C29WNY 44413525 EC50 = 30 nM T97917 CM2R4B 44413526 EC50 = 5130 nM T97917 CA3GP0 44413534 EC50 = 23 nM T97917 C9VBK6 44413547 EC50 = 310 nM T97917 CON3R2 44413548 EC50 = 81 nM T97917 C7DKA6 44413563 EC50 = 83 nM T97917 COBN46 44413564 EC50 = 100 nM T97917 CE3AU5 44413574 EC50 > 10000 nM T97917 CQ5Z1U 44413591 EC50 > 10000 nM T97917 CQKC60 44413646 EC50 = 150 nM T97917 C9RSQ3 71362579 EC50 = 19 nM T97917 C6DSX0 71525378 EC50 = 2.3 nM T97917 CC51VT 71525458 EC50 = 1 nM T97917 CDRO97 71525548 EC50 = 19315 nM T97917 C67QTG 71698362 EC50 = 1000 nM T97917 CU3K2T 71698365 EC50 = 1700 nM T97917 CYT92I 71698442 EC50 = 29400 nM T97917 CK9Q5W 71698446 EC50 > 50000 nM T97917 CNI78T 71698527 EC50 = 7700 nM T97917 C25ITN 71698528 EC50 = 5500 nM T97917 C43WJT 71698529 EC50 = 7200 nM T97917 CPJ6L3 71698530 EC50 > 50000 nM T97917 CT01IM 71698531 EC50 = 4300 nM T97917 CK8V5I 71698532 EC50 > 50000 nM T97917 C5P3LQ 71698620 EC50 > 50000 nM T97917 CUI9K5 71698621 EC50 > 50000 nM T97917 CJRV63 71698622 EC50 > 50000 nM T97917 CPO3W2 71698623 EC50 > 50000 nM T97917 C05SFZ 71698624 EC50 > 50000 nM T97917 CS2TY5 71698709 EC50 > 50000 nM T97917 C7EBU6 71698710 EC50 > 50000 nM T97917 C4F5DE 71698711 EC50 > 50000 nM T97917 C6D2NC 71698712 EC50 > 50000 nM T97917 CI4FT0 71698713 EC50 > 50000 nM T97917 CW0M1S 71698793 EC50 > 50000 nM T97917 C3ALW5 71698794 EC50 > 50000 nM T97917 C27VXB 71698795 EC50 > 50000 nM T97917 C18AYL 71698796 EC50 > 50000 nM T97917 C9XQT1 71698797 EC50 > 50000 nM T97917 CH2AN3 71698877 EC50 > 50000 nM T97917 CH03IG 71698878 EC50 > 50000 nM T97917 CBTW91 71698880 EC50 = 11600 nM T97917 C7C0AG 71698881 EC50 > 50000 nM T97917 CP1FY3 71698966 EC50 > 50000 nM T97917 CU5JI8 71698967 EC50 > 50000 nM T97917 CHZ39E 71698968 EC50 > 50000 nM T97917 C9JOI7 71698969 EC50 > 50000 nM T97917 CKOY37 71698970 EC50 > 50000 nM T97917 CW7G4H 71698971 EC50 > 50000 nM T97917 C67VPX 71698972 EC50 = 6300 nM T97917 CKY03S 71699059 EC50 = 14100 nM T97917 CU13WD 71699060 EC50 = 11400 nM T97917 CM7BJ1 71699061 EC50 > 50000 nM T97917 CF92UE 71699062 EC50 = 2800 nM T97917 CPV70F 71699063 EC50 = 27200 nM T97917 C5BET3 71699064 EC50 > 50000 nM T97917 CP01IH 71699065 EC50 > 50000 nM T97917 CO03UK 71699139 EC50 = 16900 nM T97917 CQ75GP 71699140 EC50 > 50000 nM T97917 CGJ5X6 71699141 EC50 > 50000 nM T97917 CCT6F3 71699142 EC50 = 7800 nM T97917 CT81IA 71699143 EC50 = 2800 nM T97917 CYJ18T 71699222 EC50 > 50000 nM T97917 CG68MZ 92263206 EC50 = 10500 nM T97917 CX7HU0 92881734 EC50 = 250 nM T97917 CJ6U2X 93095549 EC50 = 50 nM T97917 C7O2QZ 93095555 EC50 = 160 nM T97917 C4D0FG 93095777 EC50 = 140 nM T97917 CICJ19 98363171 EC50 = 130 nM T97917 CIQZ28 118730407 EC50 = 7500 nM T97917 C86HCX 122180577 EC50 = 140 nM T97917 C4IO1T 122180578 EC50 = 300 nM T97917 C19ZHU 122180579 EC50 = 300 nM T97917 CNL3R2 122180580 EC50 = 4 nM T97917 CKDH20 122180581 IC50 = 41 nM T97917 CP37QL 122181231 EC50 = 60 nM T97917 CDW15Q 122181232 EC50 = 230 nM T97917 CQO1F8 122181233 EC50 = 660 nM T97917 C3SHJ9 122181319 EC50 = 260 nM T97917 C0IOL4 122181320 EC50 = 270 nM T97917 C5FPZ6 122181322 EC50 = 430 nM T97917 C5GM1N 122181323 EC50 = 310 nM T97917 CY6L2V 122181324 EC50 = 860 nM T97917 CK9CT2 122181408 EC50 = 7 nM T97917 CM18HD 122181409 EC50 = 7300 nM T97917 C4Z3YV 122181410 IC50 = 6650 nM T97917 CME7B3 122181411 IC50 = 170 nM T97917 CUPH69 122181412 IC50 = 90 nM T97917 CX71MD 122487986 EC50 = 9549.93 nM T97917 C8WJ2I 134263912 IC50 = 3.4 nM T97917 C34XCH 134264089 IC50 = 4.4 nM T97917 CT1IZ4 134264414 IC50 = 3.7 nM T97917 CQLF60 134264894 IC50 = 3.6 nM T97917 CP0JW1 134265014 IC50 = 6.7 nM T97917 C3HN5O 134275888 IC50 = 27.8 nM T97917 CJ3QI7 137631898 IC50 = 13 nM T97917 C2QG1T 137632100 IC50 = 759 nM T97917 C4TI9R 137634576 IC50 = 34 nM T97917 CJD9A7 137636433 IC50 = 24 nM T97917 CNI19F 137638855 IC50 = 41 nM T97917 CK3PZ1 137639605 IC50 = 44 nM T97917 CV56OT 137639628 IC50 = 35 nM T97917 CN05UB 137644238 IC50 = 18 nM T97917 CCQ3S8 137645180 IC50 = 900 nM T97917 CLV37Y 137645526 IC50 = 28 nM T97917 C2SAK7 137647141 IC50 = 15 nM T97917 C7R5NE 137647209 IC50 = 94 nM T97917 C5V0KT 137650732 IC50 = 10 nM T97917 C7VZ2B 137651557 IC50 = 53 nM T97917 CTLM94 137653536 IC50 = 273 nM T97917 CFU2W7 137657539 IC50 = 1120 nM T97917 CV9LN3 145949892 EC50 = 120 nM T97917 CGR6M1 145951632 EC50 = 7600 nM T97917 C4ON9H 145951856 EC50 = 300 nM T97917 C1Q8YJ 145952485 EC50 = 630 nM T97917 CRX78Z 145952664 EC50 = 1700 nM T97917 CG18UM 145953127 EC50 = 2000 nM T97917 COX71H 145954612 EC50 = 110 nM T97917 CF4M2C 145955803 EC50 = 1700 nM T97917 C2X5OV 145956276 EC50 = 730 nM T97917 CX7RA0 145956361 EC50 = 330 nM T97917 CM9C4I 145956762 EC50 = 1500 nM T97917 CQ82AX 145958696 EC50 = 6500 nM T97917 CN36IR 145958736 EC50 = 190 nM T97917 CJ0B9Q 145963525 EC50 = 730 nM T97917 CU6K8I 145978177 EC50 = 1500 nM T97917 C8UY7H 146035588 EC50 = 51.29 nM T97917 C9S8JD 146035589 EC50 = 52.48 nM T97917 C7K4OV 153047597 IC50 = 0.7 nM T97917 C0O5MB 153047598 IC50 = 0.5 nM T97917 C8KM2F 155517009 IC50 = 12300 nM T97917 CD63JM 155524563 EC50 = 10900 nM T97917 CUPW45 155546686 IC50 = 3.8 nM T97917 CG5B8E 155561936 IC50 = 6.5 nM T97917 D0MU1V 727787 EC50 = 400 nM T97917 D0NL4R 91827351 IC50 = 80 nM T97917 D0R1FZ 5280914 IC50 = 1.8 nM T97917 D0WB8E 24776341 EC50 = 40.74 nM T97917 D0XF0A 443295 EC50 = 20400 nM T98691 D0V3YT 10324367 IC50 = 760 nM T98691 D0X9CH 3010818 IC50 = 3500 nM T98691 D0J6AU 10152654 Ki = 1258.93 nM T98691 D0HM5J 118253852 IC50 > 20000 nM T98691 D01LNG 10201696 IC50 = 48 nM T98691 D04ZIJ 5478883 IC50 = 800 nM T98691 D0T5PH 6918602 Ki = 0.068 nM T98691 CD3P2Z 8857 IC50 > 10000 nM T98691 CU27VZ 12050 IC50 > 100000 nM T98691 C05HLN 26030 Ki = 48000 nM T98691 CIF9A2 95706 IC50 = 6800 nM T98691 CVZP51 125190 IC50 = 50 nM T98691 C5YNV4 161091 IC50 = 2600 nM T98691 CV8A4D 163098 IC50 = 600 nM T98691 C4U5MD 202918 IC50 > 50000 nM T98691 C62DWI 231061 IC50 = 43000 nM T98691 C8OHY9 254021 IC50 = 600 nM T98691 C07JLH 404672 Ki = 8700 nM T98691 CN67CR 555078 IC50 > 100000 nM T98691 CRY54Z 690107 IC50 > 10000 nM T98691 C31BIK 832505 IC50 = 15000 nM T98691 C65UJT 980235 IC50 = 31630 nM T98691 C25SXA 1440071 IC50 = 24390 nM T98691 C9RQ2F 2848907 IC50 = 1600 nM T98691 CT8KV2 3001308 IC50 > 10000 nM T98691 CTE79D 3011892 Ki = 760000 nM T98691 C08KQP 3032999 IC50 > 10000 nM T98691 CWU18B 3082865 Ki = 1.3 nM T98691 CU43OY 3088969 Ki = 134000 nM T98691 C3G8IK 3731185 IC50 = 170 nM T98691 CKM1S9 3827422 IC50 = 510 nM T98691 CMW5A9 4430623 Ki = 245000 nM T98691 C2ZN0V 4479093 IC50 = 90000 nM T98691 CR2ND4 5287468 Ki = 2.2 nM T98691 CW6D7Z 5287498 IC50 = 160000 nM T98691 CB6H0T 5287549 Ki = 0.49 nM T98691 CESY50 5288259 IC50 = 330 nM T98691 C6YF4B 5288616 IC50 = 89 nM T98691 CFM6E4 5288618 IC50 = 82 nM T98691 C9E1UW 5288633 Ki = 700 nM T98691 CN3RY0 5289345 Ki = 340 nM T98691 CWOL57 5339865 IC50 = 45000 nM T98691 CR6B4P 5465605 IC50 > 10000 nM T98691 C3B5YE 5728928 IC50 > 100000 nM T98691 C57VBE 5762376 IC50 > 10000 nM T98691 CW94RA 5897251 IC50 = 98680 nM T98691 C3KI5C 5910205 IC50 > 10000 nM T98691 C1DAZ6 6420159 Ki > 10000 nM T98691 CD51MJ 6442675 IC50 = 30340 nM T98691 CQM64S 6610323 IC50 = 1.9 nM T98691 C0XQP7 6917747 IC50 > 100000 nM T98691 C9BGP6 7020268 Ki = 16000 nM T98691 C7WP6J 8194707 IC50 > 100000 nM T98691 CUXQ12 8832875 IC50 = 29810 nM T98691 C2GV5W 8854795 IC50 > 100000 nM T98691 CN26IL 9547980 Ki > 30000 nM T98691 CF40ZX 9562299 IC50 > 10000 nM T98691 C3QN6S 9571439 IC50 > 10000 nM T98691 CLE53W 9580655 IC50 = 741 nM T98691 CC2ZY8 9580662 IC50 = 228 nM T98691 CT3Y9G 9580665 IC50 = 369 nM T98691 CE42MQ 9809035 Ki = 28.8 nM T98691 CB32AH 9812750 IC50 = 430 nM T98691 C4UE3W 9813935 IC50 = 11500 nM T98691 CQ1NG7 9815041 IC50 = 498 nM T98691 CIX3A6 9816412 IC50 = 80 nM T98691 COBW38 9821383 IC50 = 3090 nM T98691 C9F7PL 9825191 Ki = 22300 nM T98691 C0N4DH 9825355 IC50 = 1800 nM T98691 CN51PR 9829299 Ki = 1000 nM T98691 CK7B2P 9829646 IC50 = 20 nM T98691 C2AI0Z 9834360 IC50 = 1750 nM T98691 CNU47F 9834637 IC50 = 20000 nM T98691 CLND75 9835685 IC50 = 850 nM T98691 CLQ92U 9848147 IC50 = 10000 nM T98691 C8TL5X 9855884 IC50 = 650 nM T98691 CVS7N2 9877581 IC50 = 100 nM T98691 CC3X2P 9877623 IC50 = 100 nM T98691 CO0PD1 9883178 IC50 = 300 nM T98691 CCAI25 9886751 IC50 = 15 nM T98691 C0NM3D 9887557 IC50 = 990 nM T98691 CGA91J 9890145 IC50 > 10000 nM T98691 C8P5LN 9891030 Ki = 190 nM T98691 C8HI1R 9891108 IC50 = 1400 nM T98691 C5L4YE 9893225 IC50 = 1.2 nM T98691 COK50T 9895628 IC50 = 18 nM T98691 CIBS75 9899272 IC50 = 150 nM T98691 C2JCM5 9902742 IC50 = 400 nM T98691 C5XS2F 9904539 Ki = 700 nM T98691 CALH63 9908450 IC50 = 320 nM T98691 C7WKG9 9913437 IC50 > 10000 nM T98691 C78CYD 9920989 IC50 = 23000 nM T98691 CXD2Y6 9926586 IC50 = 500 nM T98691 CNR6D5 9948720 IC50 = 55 nM T98691 C0PJ2U 9964915 IC50 = 50 nM T98691 C4WFJ2 9980678 Ki = 640 nM T98691 CBNR45 9980918 IC50 > 1000 nM T98691 CHN80D 9981917 IC50 > 10000 nM T98691 C1F4BA 9984481 IC50 = 10.7 nM T98691 C69FCE 9987052 Ki = 930 nM T98691 C7P6JO 10004326 IC50 > 1000 nM T98691 C40APB 10005577 IC50 > 1000 nM T98691 CI96RJ 10008050 IC50 = 48.7 nM T98691 CXY9N8 10024008 IC50 > 1000 nM T98691 CLB5G0 10025017 IC50 = 410 nM T98691 C4NW7I 10026902 IC50 > 1000 nM T98691 C0SJY5 10031327 IC50 = 139 nM T98691 C68HGW 10047261 IC50 = 352 nM T98691 C8F7MU 10047536 IC50 > 1000 nM T98691 C2N9CS 10062713 IC50 = 12 nM T98691 C1QB5U 10063343 IC50 = 2900 nM T98691 C5KR4U 10068161 IC50 = 4300 nM T98691 C1IZ3A 10075688 Ki = 0.6 nM T98691 CV29YC 10076076 IC50 = 1700 nM T98691 CHA42Q 10097070 IC50 > 10000 nM T98691 CD6L1T 10098422 Ki = 19 nM T98691 C8FPB5 10098917 IC50 = 1 nM T98691 CSO9B2 10099774 Ki = 120 nM T98691 CA5N3E 10111943 IC50 = 115 nM T98691 C57JDN 10118049 IC50 = 11.5 nM T98691 CFC3Q8 10120133 IC50 = 33000 nM T98691 C6AZ3B 10120903 IC50 = 1000000 nM T98691 C97NJR 10121949 Ki = 11000 nM T98691 C7XOA0 10127183 IC50 = 344 nM T98691 CSO96K 10127748 IC50 = 1300 nM T98691 CKZ15P 10129236 IC50 = 680 nM T98691 CJ79ZX 10138553 IC50 = 1667 nM T98691 CY6PU1 10143615 Ki = 3.9 nM T98691 CLID02 10144235 Ki = 19000 nM T98691 CQ3YD8 10150891 IC50 = 1475 nM T98691 C8DQG0 10154619 IC50 > 10000 nM T98691 C9VFI4 10161284 IC50 = 24000 nM T98691 C1Q2EX 10164497 Ki = 300 nM T98691 CDX7R4 10164961 IC50 = 17000 nM T98691 C5B1HM 10165557 IC50 = 10000 nM T98691 C09ALX 10165785 Ki = 0.04 nM T98691 CR62PT 10165786 Ki = 52 nM T98691 CTJ7R3 10166544 IC50 = 36000 nM T98691 CDRE91 10167323 Ki = 37000 nM T98691 CZ1A8U 10173731 IC50 = 524 nM T98691 C5NEX6 10174161 IC50 = 2200 nM T98691 C1YR4T 10174359 IC50 = 1300 nM T98691 CD4G7F 10179450 IC50 = 108 nM T98691 CTON03 10179451 IC50 = 2101 nM T98691 C07GUT 10184761 Ki = 390 nM T98691 C4M3SG 10186046 IC50 = 3800000 nM T98691 CCO7A6 10187105 Ki = 10000 nM T98691 CP2M1T 10187189 Ki = 4.2 nM T98691 C9WTI5 10187190 Ki = 45 nM T98691 C0SF7U 10187920 IC50 = 10000 nM T98691 CKZ1A0 10194354 IC50 = 80 nM T98691 CZD7A6 10194447 IC50 = 878 nM T98691 CA2UH4 10194634 IC50 = 887 nM T98691 CO7XD6 10198366 IC50 = 6 nM T98691 C5T8PK 10198752 IC50 = 54 nM T98691 CQ8YM3 10199981 Ki = 9600 nM T98691 CL9DW3 10200425 IC50 = 4804 nM T98691 CS3IP7 10210867 IC50 = 190000 nM T98691 C1WL9J 10211340 Ki = 1400 nM T98691 CV0CI4 10216098 Ki = 20 nM T98691 C1F9SP 10216231 IC50 = 1857 nM T98691 C1Y3QZ 10216510 IC50 = 1670 nM T98691 C5GSN6 10216511 IC50 = 2792 nM T98691 CT8K5D 10231379 IC50 = 8700 nM T98691 C4OZ5K 10231447 IC50 = 69000 nM T98691 CJBI61 10237771 IC50 = 13 nM T98691 CFI43Z 10238903 IC50 = 470 nM T98691 CORW86 10247897 IC50 = 150 nM T98691 CEQ21I 10249499 IC50 > 1000 nM T98691 C6A8NV 10252643 Ki = 81 nM T98691 C9SOH2 10271564 IC50 = 1682 nM T98691 CKX0R7 10287617 IC50 = 34 nM T98691 CUW38E 10288162 IC50 = 1001 nM T98691 CX23AL 10288163 IC50 = 3002 nM T98691 CY7DQ2 10288811 IC50 = 1600 nM T98691 CV9LB1 10302710 IC50 = 17000 nM T98691 CUQ2R3 10303526 IC50 = 240000 nM T98691 CV5S7B 10303657 IC50 = 1000000 nM T98691 CZR02J 10303878 Ki = 7500 nM T98691 CPT49O 10310362 IC50 = 3047 nM T98691 CO0GQ8 10313520 IC50 = 450 nM T98691 C9DN6G 10325113 IC50 = 31.9 nM T98691 CXN4D2 10327819 Ki = 70 nM T98691 C59ZDR 10337631 IC50 > 1000 nM T98691 C2GLK6 10346121 IC50 = 0.1 nM T98691 C7D9XB 10363069 IC50 = 22000 nM T98691 CDY26B 10366413 Ki = 6100 nM T98691 CDX2C8 10367993 IC50 > 1000 nM T98691 CYF98Z 10368089 IC50 = 2300 nM T98691 CD9ZI0 10373289 Ki = 720 nM T98691 CX7S8A 10392779 IC50 = 10.8 nM T98691 C7LU1Z 10395274 Ki = 74000 nM T98691 CF7O6A 10409137 IC50 > 20000 nM T98691 C41JUO 10414118 IC50 = 3.8 nM T98691 CDVZ19 10431266 Ki = 6800 nM T98691 CCD1B8 10433014 IC50 = 7 nM T98691 C8DTH3 10436731 IC50 = 554 nM T98691 C57DYJ 10437715 Ki = 2 nM T98691 CN18SE 10456222 Ki = 0.47 nM T98691 C06QJW 10457653 IC50 = 0.1 nM T98691 CK9PX5 10461097 Ki > 1000 nM T98691 C6KJM2 10461790 Ki = 154000 nM T98691 C5M7BL 10471316 IC50 = 1000 nM T98691 CXD68E 10473874 IC50 = 190 nM T98691 C32MAD 10482525 IC50 < 0.4 nM T98691 CW7V0M 10496067 IC50 > 1000 nM T98691 C1MX2S 10499322 Ki = 250 nM T98691 CHTL13 10507714 Ki = 39 nM T98691 CZ80TL 10507960 Ki > 1000 nM T98691 CGA7D1 10515827 IC50 = 350 nM T98691 C25HQJ 10522795 Ki > 1000 nM T98691 C0UBF5 10524384 Ki = 580 nM T98691 CZUA37 10531571 Ki > 1000 nM T98691 COP6I9 10566003 IC50 = 200 nM T98691 CR54HQ 10569603 Ki > 10000 nM T98691 C8U1RQ 10593841 Ki = 2600 nM T98691 CM29WH 10663100 IC50 = 290 nM T98691 CJ7U3O 10668284 IC50 > 10000 nM T98691 CRL23A 10674588 Ki > 1000 nM T98691 C9PY4N 10690022 Ki = 850 nM T98691 CKO6L0 10698950 Ki = 16 nM T98691 CP2WG8 10716501 IC50 = 32 nM T98691 C5E8FN 10793407 Ki = 290 nM T98691 C9AIY1 10793962 Ki = 49 nM T98691 C9XI7T 10804795 IC50 = 900 nM T98691 CQ08YK 10807774 Ki > 1000 nM T98691 CHC3F0 10817683 Ki = 290 nM T98691 CZ4V0F 10832380 Ki > 10000 nM T98691 C78VEK 10837067 Ki > 1000 nM T98691 C1BT8R 10853144 IC50 = 110 nM T98691 CBWJ85 10862359 IC50 = 6273 nM T98691 CNVG58 10875013 IC50 > 10000 nM T98691 CMO9Y1 10886114 Ki = 9.6 nM T98691 C7ZNC2 10892596 IC50 = 170 nM T98691 CZK49P 10893343 IC50 = 2710 nM T98691 CBJ1I7 10902914 IC50 > 10000 nM T98691 CA30HS 10905508 IC50 > 10000 nM T98691 CA9ZC6 10907387 Ki = 44 nM T98691 C5X6NA 10924832 IC50 = 5583 nM T98691 CZG37Y 10938664 IC50 > 10000 nM T98691 CA72YH 10949332 IC50 = 31 nM T98691 CL7W4P 10960628 IC50 = 800 nM T98691 CW1L5K 10960899 IC50 = 1500 nM T98691 CR0P8J 10971179 IC50 > 10000 nM T98691 CK9E8W 10972182 IC50 = 3907 nM T98691 C6ZOI1 10979734 IC50 = 5952 nM T98691 CCFA87 10983274 IC50 = 80 nM T98691 CA3NG9 10993428 IC50 > 10000 nM T98691 C7BI2T 11009218 IC50 = 2600 nM T98691 CM9Z5T 11012257 IC50 = 825 nM T98691 C5XHI0 11014664 IC50 = 1593 nM T98691 C56FMI 11027472 Ki = 7.9 nM T98691 CL19TE 11028356 Ki = 2.8 nM T98691 CY72BF 11034349 IC50 > 10000 nM T98691 CQXP76 11050104 Ki = 144.4 nM T98691 CMP6K1 11071803 Ki = 4.7 nM T98691 CY3V4J 11080121 IC50 = 6 nM T98691 C0PSR8 11081485 IC50 > 10000 nM T98691 C5WY1H 11082075 IC50 < 30 nM T98691 CMC63T 11113842 Ki = 28.8 nM T98691 CQ4L0T 11122768 IC50 = 50 nM T98691 CQK6U4 11144121 IC50 = 4000 nM T98691 CDR7A6 11155973 Ki = 24 nM T98691 C8EAL0 11156785 Ki = 193 nM T98691 C9SN1Q 11157631 Ki = 98 nM T98691 CH41OF 11157632 Ki = 1520 nM T98691 C61AIQ 11168385 Ki = 588 nM T98691 CAI94Q 11168613 Ki = 372 nM T98691 C2VJG7 11178623 Ki = 541 nM T98691 CMDU74 11180007 Ki = 11530 nM T98691 CS90MB 11191512 Ki = 2678 nM T98691 CN0F8E 11199915 IC50 = 1270 nM T98691 C2H4GP 11200735 Ki = 11 nM T98691 CTCX89 11203484 Ki > 65000 nM T98691 C17UIX 11203679 IC50 = 560 nM T98691 C7SOL0 11224927 Ki = 7460 nM T98691 CM8ZV1 11225780 Ki = 18900 nM T98691 CLC2X1 11226457 Ki = 1800 nM T98691 C0JO5R 11238059 Ki > 100000 nM T98691 C3T1LM 11238468 Ki > 50000 nM T98691 C5VY1E 11247716 Ki = 9040 nM T98691 CLA6J3 11249688 Ki > 37000 nM T98691 CRXU26 11250282 Ki = 2310 nM T98691 CHK9N2 11261516 Ki = 3520 nM T98691 C8F2ZN 11269453 IC50 > 1000 nM T98691 CIFQ06 11273375 Ki = 5 nM T98691 C15XUE 11283547 Ki = 11530 nM T98691 CCH6N4 11283555 IC50 = 456 nM T98691 CM86BP 11294094 Ki = 11800 nM T98691 CFU50G 11294227 Ki = 2830 nM T98691 CV86IB 11295906 Ki > 11000 nM T98691 CZX89I 11305296 Ki = 8370 nM T98691 CR2T5B 11305867 Ki = 914 nM T98691 CU6Z0F 11306593 Ki > 37000 nM T98691 CEC0A2 11316876 Ki > 10000 nM T98691 CDYL91 11327594 Ki > 100000 nM T98691 CP5MI6 11329727 Ki > 30000 nM T98691 CD70PA 11341599 Ki = 108 nM T98691 C5X1VW 11351327 IC50 = 62 nM T98691 CFJ70U 11353015 Ki = 4670 nM T98691 C9W0TB 11375856 Ki > 100000 nM T98691 C7NQX3 11375955 Ki = 777 nM T98691 CH4I3T 11375956 IC50 = 230 nM T98691 C34DFQ 11376188 Ki > 70000 nM T98691 CAL7B2 11376611 Ki > 100000 nM T98691 COV1F4 11387157 Ki = 48370 nM T98691 CEW0F3 11387421 Ki = 4080 nM T98691 C3DQL2 11396020 Ki > 30000 nM T98691 C4QM7I 11396148 Ki > 10000 nM T98691 CER2V8 11397519 Ki = 1730 nM T98691 C4ZLU9 11397590 Ki > 30000 nM T98691 C7RFC5 11398171 Ki = 267 nM T98691 CI3HK2 11409407 Ki = 849 nM T98691 CO4Y3H 11410560 Ki > 100000 nM T98691 CU4P8A 11418931 Ki = 17 nM T98691 C56SXA 11419952 Ki = 1150 nM T98691 CGD1K4 11421700 Ki = 17700 nM T98691 CILJ37 11431699 Ki > 30000 nM T98691 CM2VQ6 11431993 Ki = 9670 nM T98691 C19YRB 11432272 Ki = 8990 nM T98691 C72PFO 11432501 Ki = 123 nM T98691 C65ASH 11432773 Ki > 100000 nM T98691 CQRB45 11433280 Ki = 636 nM T98691 CQIP48 11439739 IC50 = 76 nM T98691 CH9ZA7 11443990 Ki = 199 nM T98691 C1AT2Z 11453155 IC50 = 68 nM T98691 CL53MS 11456165 Ki > 100000 nM T98691 CME32S 11456379 Ki > 100000 nM T98691 C0O8MK 11464526 IC50 = 44 nM T98691 C5N3BV 11466327 Ki > 10000 nM T98691 CV43WB 11466677 Ki = 285 nM T98691 CM59AQ 11466845 Ki = 1180 nM T98691 CL1D2Z 11471738 IC50 = 1711 nM T98691 C0ZK5I 11477975 Ki = 150 nM T98691 C9U0YI 11478637 Ki = 3936 nM T98691 CBC8U6 11490230 Ki = 369 nM T98691 CM41QW 11494775 Ki = 54 nM T98691 CT8S4U 11496335 Ki = 900 nM T98691 C5CL9A 11496988 Ki > 15000 nM T98691 CC92RV 11501571 IC50 = 32000 nM T98691 CFI8L5 11502586 IC50 = 150 nM T98691 CK5JM6 11503223 IC50 = 2274 nM T98691 CY4A7V 11504785 Ki = 5 nM T98691 C3Q7BE 11504819 Ki = 150 nM T98691 CCH09G 11507712 Ki > 150000 nM T98691 CHI9N5 11512144 Ki = 8800 nM T98691 C23DKS 11516307 IC50 > 10000 nM T98691 CDA9F5 11517167 Ki > 150000 nM T98691 C6D2VI 11525733 Ki = 2000 nM T98691 CW4ED1 11532268 IC50 = 120 nM T98691 CQ69XF 11533114 Ki = 12000 nM T98691 C2BT3L 11533910 Ki > 150000 nM T98691 C98EQF 11545899 IC50 = 540 nM T98691 C6XK8V 11547772 Ki = 8900 nM T98691 CG57TI 11551229 Ki > 150000 nM T98691 CXTQ39 11558838 Ki = 88000 nM T98691 CF9DE7 11561418 Ki = 71000 nM T98691 CA61ZJ 11562424 Ki = 11000 nM T98691 CKH13D 11562461 Ki = 9100 nM T98691 CTN57Q 11562607 Ki = 1600 nM T98691 CB3W8O 11565199 Ki = 1540 nM T98691 CPY84F 11569750 Ki = 430 nM T98691 CW1O0M 11569883 Ki = 1200 nM T98691 C1TV6S 11580329 Ki = 25000 nM T98691 C73VCU 11584899 Ki = 1.7 nM T98691 CJG6T3 11585276 Ki = 0.57 nM T98691 CER65Q 11588182 Ki = 430 nM T98691 CUX70T 11588744 Ki > 150000 nM T98691 C2Y6JE 11590993 Ki = 2300 nM T98691 CLV84W 11594784 Ki > 150000 nM T98691 C1QO2C 11598043 IC50 = 180 nM T98691 C85WBA 11599792 Ki = 400 nM T98691 CQZ5T4 11602113 Ki > 5000 nM T98691 C1NV2U 11605163 Ki = 11000 nM T98691 CM4OS2 11606272 Ki = 1.4 nM T98691 C98KMP 11612451 Ki = 2200 nM T98691 CZU5E4 11613136 Ki = 8800 nM T98691 CK0AN9 11616537 Ki = 18000 nM T98691 CE8WO5 11618337 Ki = 3200 nM T98691 CTL1P3 11618795 Ki = 420 nM T98691 CQ7KD1 11623853 Ki = 23000 nM T98691 C9LBF3 11628054 Ki = 160 nM T98691 CUS5Q4 11630803 Ki = 45000 nM T98691 C70VTY 11631953 Ki = 7900 nM T98691 C98QKS 11635243 Ki = 7.9 nM T98691 CLMY50 11641509 Ki = 7600 nM T98691 CILB73 11649751 Ki > 17000 nM T98691 CJRN14 11655672 Ki = 15000 nM T98691 C5ZOM0 11656060 IC50 = 16 nM T98691 C0Q7AH 11662896 Ki = 5600 nM T98691 C4YFI9 11663730 IC50 = 10 nM T98691 C0D7NS 11663810 Ki = 16000 nM T98691 C5SJ9K 11669355 IC50 > 10000 nM T98691 C13TGX 11671560 Ki = 540 nM T98691 CT0OZ8 11673881 Ki = 37000 nM T98691 C1BGL5 11677886 Ki = 6400 nM T98691 C23ZVP 11678241 Ki = 8.2 nM T98691 C27LJY 11678922 Ki = 0.43 nM T98691 CDNH37 11680631 Ki > 150000 nM T98691 C1Q2OT 11682028 Ki = 23000 nM T98691 C6Q8KO 11682184 Ki = 5900 nM T98691 CNB67S 11684874 Ki = 12000 nM T98691 CL4XB1 11685284 Ki = 4.5 nM T98691 C53OYX 11692372 Ki = 0.63 nM T98691 C38REW 11695166 Ki > 150000 nM T98691 CJB3E9 11695584 Ki = 48000 nM T98691 C0OC5V 11696208 Ki = 22000 nM T98691 CHP6U3 11699298 Ki = 15000 nM T98691 C7QIP8 11699507 Ki = 10 nM T98691 CRTS62 11703216 Ki = 290 nM T98691 C5UEI7 11703527 IC50 = 6760 nM T98691 C9X6PV 11703830 Ki = 88 nM T98691 CU57OC 11705307 IC50 = 83.7 nM T98691 C0Y5XV 11705688 Ki = 19000 nM T98691 C5FZ1J 11710873 IC50 = 10000 nM T98691 C26RZY 11717535 Ki = 17000 nM T98691 CDS4P0 11743922 Ki = 17 nM T98691 C0SV2T 11753412 Ki = 1490 nM T98691 CY63BP 11761693 IC50 = 90 nM T98691 C8EZR3 11763189 Ki = 1.7 nM T98691 CGU6I7 11767007 Ki = 1.5 nM T98691 C8D7BS 11771234 IC50 > 10000 nM T98691 CT5B1S 11784942 Ki > 33750 nM T98691 CDJH89 11811557 IC50 = 4641 nM T98691 CZ1YB3 11824245 IC50 > 10000 nM T98691 CRXO59 11857300 IC50 = 132 nM T98691 CDOG76 11857302 IC50 = 249 nM T98691 C5NR3L 11962098 IC50 = 83 nM T98691 C3QN1E 11983275 Ki = 1000 nM T98691 C3JO1P 12262704 IC50 > 50000 nM T98691 CP4H9E 12737307 Ki = 122000 nM T98691 C6JS5Y 13184126 Ki > 100000 nM T98691 C31MCN 13186896 IC50 > 100000 nM T98691 CA78NJ 13386706 Ki = 14000 nM T98691 C9WC6M 14655218 Ki = 230 nM T98691 C0XI2R 15296015 IC50 = 3 nM T98691 CLGV32 15547238 IC50 = 42 nM T98691 C2QO1B 15955412 Ki = 123000 nM T98691 CHC31Q 15985697 IC50 = 667 nM T98691 C9LW6H 15985754 IC50 = 67 nM T98691 CQ5F9T 16045426 IC50 = 0.7 nM T98691 CL38RU 16046125 Ki > 100000 nM T98691 CQ2N8D 16046128 Ki = 3120 nM T98691 CY0FX8 16061496 IC50 = 574 nM T98691 C08XJK 16090559 Ki > 10000 nM T98691 CTIV96 16090560 Ki > 10000 nM T98691 C2QWA9 16090561 Ki > 10000 nM T98691 CJBT92 16090562 Ki > 10000 nM T98691 CU6KB8 16090563 Ki > 15000 nM T98691 CZ9J6G 16108888 IC50 = 0.17 nM T98691 C3KMJ0 16108889 IC50 = 5.1 nM T98691 CM7DA6 16108890 IC50 = 0.34 nM T98691 C0M1KY 16108891 IC50 = 1.2 nM T98691 C63XFT 16108892 IC50 = 3.9 nM T98691 C0LJ8Y 16108893 IC50 = 0.33 nM T98691 C7IQ0W 16108894 IC50 = 0.52 nM T98691 CPN5S2 16108895 IC50 = 0.58 nM T98691 CJ98LN 16108900 IC50 = 1.1 nM T98691 CYT2X8 16108901 IC50 = 0.31 nM T98691 CJRB12 16108902 IC50 = 0.45 nM T98691 C0QAC5 16108903 IC50 > 10 nM T98691 CT65ZO 16108904 IC50 = 0.82 nM T98691 CHKR18 16108905 IC50 = 1.7 nM T98691 CZI27Q 16108906 IC50 = 0.68 nM T98691 C5FUL9 16661369 IC50 = 63060 nM T98691 CUTI57 16661526 IC50 = 55728 nM T98691 C26JIW 16661682 IC50 = 17043 nM T98691 C6XPN4 16664855 IC50 = 22 nM T98691 C8XLP2 16720100 Ki > 15000 nM T98691 C4P8ZV 16720327 Ki = 5190 nM T98691 C7Y6EF 16725315 IC50 = 56 nM T98691 CKA87T 17945762 IC50 = 42 nM T98691 CH4TC1 17968209 IC50 > 1000 nM T98691 C0JBH9 18395047 IC50 = 780 nM T98691 C2XTI9 18395048 IC50 = 91 nM T98691 C7WD4Z 18628647 IC50 = 8391 nM T98691 CR7B9L 18628679 IC50 > 10000 nM T98691 CHA0S3 18628693 IC50 = 2755 nM T98691 CU3NM9 18628717 IC50 > 10000 nM T98691 C71IFZ 18628739 IC50 = 9546 nM T98691 CUSD12 18628799 IC50 = 140 nM T98691 C5ZRU1 19540655 IC50 > 100000 nM T98691 CLM2E4 19959068 IC50 = 37000 nM T98691 CP1A6L 20262575 IC50 = 7200 nM T98691 C8O5CM 20828112 Ki = 28000 nM T98691 C2KBL6 22972497 IC50 > 10000 nM T98691 CD5R3V 22972573 IC50 = 2235 nM T98691 CFY7O6 22988664 Ki = 182000 nM T98691 CKW6Q8 23626706 IC50 = 230 nM T98691 CS0G9W 23631927 IC50 = 7 nM T98691 C0QVL2 23644739 Ki = 20 nM T98691 CM1C8V 23644740 Ki = 380 nM T98691 CM5TI6 23644741 Ki = 5040 nM T98691 CMQ72V 23644742 Ki > 100000 nM T98691 CZPF48 23648277 IC50 = 430 nM T98691 CHU59C 23648278 IC50 = 456 nM T98691 CA74XT 23648279 IC50 > 10000 nM T98691 C2I6RW 23648280 IC50 > 10000 nM T98691 CCJ8M5 23648281 IC50 > 10000 nM T98691 C9C0HK 23648282 IC50 = 911 nM T98691 CC50JD 23648283 IC50 = 1035 nM T98691 CS1VW7 23648284 IC50 = 86 nM T98691 CUQH43 23648285 IC50 = 105 nM T98691 CM52JD 23648286 IC50 = 121 nM T98691 CE09VM 23648287 IC50 > 10000 nM T98691 C1FRI4 23648288 IC50 > 10000 nM T98691 C9RNB7 23648289 IC50 = 22 nM T98691 C4J5MD 23648290 IC50 = 15 nM T98691 CY20DH 23648291 IC50 = 23 nM T98691 CF7O3H 23648292 IC50 = 181 nM T98691 CKI1W5 23648293 IC50 = 114 nM T98691 CN5S3K 23648294 IC50 = 24 nM T98691 CTB69E 23648295 IC50 = 41 nM T98691 C31XJH 23648296 IC50 = 7 nM T98691 C5ECI8 23648297 IC50 > 10000 nM T98691 CB7T3I 23648298 IC50 = 1950 nM T98691 CVF2M6 23648299 IC50 = 34 nM T98691 CRZ56K 23648300 IC50 = 1473 nM T98691 CQ1C8H 23648301 IC50 = 809 nM T98691 CQFD10 23648302 IC50 = 560 nM T98691 CFR23Q 23648303 IC50 = 1480 nM T98691 C0FBS2 23648304 IC50 = 771 nM T98691 C67AYX 23648305 IC50 = 1915 nM T98691 CN6R9M 23648306 IC50 = 314 nM T98691 C85PXH 23648308 IC50 = 2422 nM T98691 CVH82R 23648309 IC50 = 342 nM T98691 COZK65 23648310 Ki = 7 nM T98691 CCF89E 23648311 Ki = 216 nM T98691 CS4NV6 23648312 Ki = 22 nM T98691 CC9S7T 23648313 Ki = 4.6 nM T98691 CCTK94 23648314 Ki = 326 nM T98691 CG29HR 23648315 Ki = 134 nM T98691 CY35VT 23648316 Ki = 3.7 nM T98691 CTX79K 23648317 Ki = 1.4 nM T98691 C8T5FW 23648318 Ki = 1.5 nM T98691 C02UQZ 23648319 Ki = 5 nM T98691 C1QVI4 23648320 Ki = 3.4 nM T98691 CP4SY0 23648321 Ki = 2.8 nM T98691 C9C7JR 23648322 Ki = 9.3 nM T98691 CTY4J2 23648323 Ki = 23 nM T98691 CGJ96H 23648326 Ki = 2991 nM T98691 CSI84Q 23648327 Ki = 4214 nM T98691 C2PD6A 23648328 Ki = 1.1 nM T98691 C37FRY 23648329 Ki = 7.2 nM T98691 C4KU8Q 23648330 Ki = 1.2 nM T98691 C09TQZ 23648331 Ki = 25 nM T98691 CM0AG6 23648332 Ki = 13 nM T98691 C8DJZ7 23648333 Ki = 68 nM T98691 CVH46G 23648334 Ki = 14 nM T98691 C1IRW9 23648335 Ki > 79000 nM T98691 CWG7T3 23648336 Ki = 106 nM T98691 CZN75B 23648337 Ki > 37000 nM T98691 CLZX16 23648338 Ki = 148 nM T98691 C5UDE3 23648339 Ki = 303 nM T98691 C7V6EY 23648340 Ki = 176 nM T98691 CRK1M0 23648341 Ki = 7950 nM T98691 C34VFB 23648342 Ki = 1296 nM T98691 CQUD83 23648343 Ki = 316 nM T98691 C32GYK 23648344 Ki > 6440 nM T98691 CHQ82B 23648345 Ki = 14 nM T98691 CH0XM8 23648346 Ki = 120 nM T98691 C8ZT0W 23648347 Ki = 92 nM T98691 C5T6WQ 23648348 Ki = 62 nM T98691 CKE2C0 23648349 Ki = 88 nM T98691 CUH90V 23648350 Ki = 9200 nM T98691 CCA45G 23648351 Ki = 2 nM T98691 CP10ST 23648352 Ki = 15530 nM T98691 CZRA72 23648353 Ki = 1800 nM T98691 CPTK56 23648354 Ki = 20 nM T98691 C1YMU6 23648355 Ki = 19 nM T98691 C58JSH 23648356 Ki = 42 nM T98691 C5YS0D 23648357 Ki = 3410 nM T98691 CNHA15 23648358 Ki = 1.6 nM T98691 CQVC57 23648359 Ki = 75 nM T98691 C03ZCQ 23648360 Ki > 30000 nM T98691 CM5QI0 23648361 Ki > 100000 nM T98691 C6YRH9 23648362 Ki > 100000 nM T98691 CP6Q2L 23648363 Ki > 100000 nM T98691 C63OZA 23648364 Ki > 100000 nM T98691 COU98B 23648365 Ki = 8860 nM T98691 CK43WQ 23648366 Ki = 197 nM T98691 CKQ0P4 23648367 Ki > 30000 nM T98691 CGSN32 23648368 Ki > 100000 nM T98691 C76JKU 23648369 Ki > 100000 nM T98691 C46RQB 23648370 Ki > 30000 nM T98691 CPC7Z2 23648371 Ki > 30000 nM T98691 C5FJZ6 23648372 Ki > 100000 nM T98691 CL8X1T 23648373 Ki > 100000 nM T98691 CL01QA 23648374 Ki = 5470 nM T98691 CG9N8B 23648375 Ki = 6030 nM T98691 CT98GY 23648376 Ki = 9790 nM T98691 CX6JF9 23648377 Ki > 100000 nM T98691 CJ7N9D 23648378 Ki > 100000 nM T98691 C0GQ4R 23648379 Ki > 30000 nM T98691 CYS7Z2 23648380 Ki > 30000 nM T98691 C6H3DY 23648381 Ki > 100000 nM T98691 CGV2J8 23648382 Ki > 100000 nM T98691 CF0JM1 23648383 Ki > 100000 nM T98691 C5LGJ7 23648384 Ki > 100000 nM T98691 C39FZB 23648385 Ki > 100000 nM T98691 C85STC 23648386 Ki > 100000 nM T98691 CWV98T 23648387 Ki > 100000 nM T98691 CX59EJ 23648388 Ki > 100000 nM T98691 CFNX14 23648389 Ki > 100000 nM T98691 CZC34G 23648390 Ki > 100000 nM T98691 C1FJY7 23648391 Ki = 4970 nM T98691 C9KW2O 23648392 Ki = 45 nM T98691 CI58TU 23648393 Ki = 7940 nM T98691 CB3JX0 23648394 Ki = 582 nM T98691 CYBW67 23648395 Ki = 331 nM T98691 CR1K4V 23648396 Ki = 4790 nM T98691 C1B9GH 23648397 Ki = 594 nM T98691 CF72ZM 23648398 Ki = 2570 nM T98691 C9X3TS 23648399 Ki = 232 nM T98691 CL8RT9 23648400 Ki = 75 nM T98691 CPEW28 23648401 Ki = 125 nM T98691 CT10OV 23648402 Ki = 6 nM T98691 CEC70K 23648403 Ki = 4 nM T98691 CE2QR4 23648404 Ki = 2110 nM T98691 C4F2BY 23648405 Ki > 100000 nM T98691 CX37JK 23648406 Ki > 30000 nM T98691 CD8JP5 23648407 Ki = 14600 nM T98691 CC7HD5 23648408 Ki = 2590 nM T98691 CWGL69 23648409 Ki = 512 nM T98691 CA2DE6 23648410 Ki = 1060 nM T98691 C3VT9K 23648411 Ki = 810 nM T98691 CBR76L 23648414 IC50 = 9900 nM T98691 CZ7ME6 23648415 IC50 = 7700 nM T98691 CVU01O 23648416 IC50 = 1100 nM T98691 C3M5GX 23648417 IC50 = 1400 nM T98691 CG9NQ8 23648418 IC50 > 10000 nM T98691 C2F1MC 23648419 IC50 = 8000 nM T98691 CCZ4J1 23648420 IC50 = 2800 nM T98691 CC2W3A 23648421 IC50 = 1700 nM T98691 C8Z5BC 23648422 IC50 = 1200 nM T98691 CVD5Y6 23648423 IC50 = 330 nM T98691 CL4Q2D 23648424 IC50 < 30 nM T98691 CF0TY4 23648425 IC50 = 190 nM T98691 CX0V8M 23648426 IC50 = 154 nM T98691 CME4Y9 23648427 IC50 = 110 nM T98691 C4AJB0 23648428 IC50 = 660 nM T98691 C7DBS2 23648441 Ki = 513 nM T98691 CWY87K 23648448 IC50 = 110 nM T98691 C1YTO9 23648449 IC50 > 10000 nM T98691 CJO2P4 24776563 IC50 = 6680 nM T98691 CR8L2N 24776564 IC50 = 13550 nM T98691 C3U0QR 24776565 IC50 = 4150 nM T98691 CV9F0D 24776566 IC50 > 30000 nM T98691 COZ5C9 24776567 IC50 = 9620 nM T98691 C28RDA 24776568 IC50 > 30000 nM T98691 C9KHL2 24776569 IC50 = 14860 nM T98691 CA4KQ3 24776683 IC50 = 420 nM T98691 C92NZG 24776926 IC50 = 2530 nM T98691 CN1R6S 24776927 IC50 = 3790 nM T98691 CT06JY 24776928 IC50 = 28440 nM T98691 CHF5Y7 24776929 IC50 > 30000 nM T98691 CO3W9N 24776931 IC50 = 3910 nM T98691 C2Y8JF 24776932 IC50 > 30000 nM T98691 CPBT05 24777048 IC50 = 5060 nM T98691 CM4KX2 24777049 IC50 > 30000 nM T98691 C6ACK9 24777050 IC50 = 17100 nM T98691 CCP4V6 24777300 IC50 = 28910 nM T98691 C8JR9Q 24777301 IC50 = 300 nM T98691 CYMF31 24777302 IC50 = 1820 nM T98691 CA04CB 24777303 IC50 = 300 nM T98691 CJ3N1A 24777429 IC50 = 800 nM T98691 CBI96T 24777430 IC50 = 780 nM T98691 CAF5Y4 24777431 IC50 = 500 nM T98691 CB96XZ 24778049 IC50 = 3300 nM T98691 CK74OH 24778050 IC50 = 23280 nM T98691 CQHR89 24778051 IC50 > 30000 nM T98691 CUG91O 24778054 IC50 = 4000 nM T98691 CF30JZ 24778183 IC50 = 10520 nM T98691 CB50GN 24778184 IC50 = 10520 nM T98691 CUP2D4 24778185 IC50 = 13370 nM T98691 C15VPF 24778187 IC50 = 13550 nM T98691 CFWK93 24778188 IC50 > 30000 nM T98691 CF9WJ1 24778189 IC50 = 17140 nM T98691 CVS50O 24778317 IC50 > 30000 nM T98691 CC4TG6 24778318 IC50 = 8050 nM T98691 CTV8S9 24778319 IC50 = 5860 nM T98691 CYP8K1 24778320 IC50 = 2270 nM T98691 CPT6I2 24778321 IC50 = 10790 nM T98691 CKP1F7 24778322 IC50 > 30000 nM T98691 CB64RJ 24778323 IC50 = 6840 nM T98691 C7U5ZK 24778439 IC50 = 2280 nM T98691 CEP4D9 24778440 IC50 = 1170 nM T98691 CH8YB7 24778441 IC50 = 12940 nM T98691 CYCD75 24778442 IC50 = 26920 nM T98691 CB3K0R 24778443 IC50 > 30000 nM T98691 CQ80SX 24778444 IC50 = 610 nM T98691 CV5P1B 24778445 IC50 > 30000 nM T98691 CMI4L3 24800875 Ki = 21900 nM T98691 CAXQ09 24801230 Ki = 13500 nM T98691 CT1A2Z 24801231 Ki = 7000 nM T98691 CN0VA7 24822701 IC50 = 5400 nM T98691 C2GQ6X 24897809 Ki = 0.9 nM T98691 CZ21HD 24898027 Ki = 0.16 nM T98691 CQU38W 24900755 IC50 = 1270 nM T98691 C2S8VB 24901099 IC50 = 26 nM T98691 CIN28B 24901100 IC50 = 263 nM T98691 CD2EH0 24901101 IC50 = 230 nM T98691 CS7B3F 24901102 IC50 = 5816 nM T98691 CG9H6V 25008106 IC50 > 1000 nM T98691 CK7BR0 25023784 IC50 = 5200 nM T98691 CZH87T 25023785 IC50 = 6800 nM T98691 C2PUY3 25023786 IC50 > 1000 nM T98691 CFQM73 25023787 IC50 > 1000 nM T98691 CTK09I 25023788 IC50 = 2300 nM T98691 CDL98C 25023789 IC50 > 1000 nM T98691 CCP3G0 25023790 IC50 > 2000 nM T98691 CGI0U2 25023791 IC50 = 6200 nM T98691 CO72TX 25027584 IC50 = 280 nM T98691 C8CIY2 25030810 IC50 = 1200 nM T98691 CMS0L3 25052748 IC50 > 1000 nM T98691 C7J3MN 25053851 IC50 > 1000 nM T98691 C43JRI 25066441 IC50 = 10.1 nM T98691 C19GML 25071954 IC50 = 150 nM T98691 CF54QZ 25129041 IC50 > 100000 nM T98691 CDO26T 25129042 IC50 > 7943.28 nM T98691 C57LJM 25129043 IC50 > 10000 nM T98691 C3AT6W 25130088 IC50 > 10000 nM T98691 C1FWI6 25133836 IC50 > 10000 nM T98691 CYV1J6 25133837 IC50 > 10000 nM T98691 CBZK08 25133838 IC50 > 50118.72 nM T98691 CUC8N5 25141405 IC50 > 100000 nM T98691 CP8U3Q 25142042 IC50 > 40000 nM T98691 C3C8YJ 25174148 IC50 = 501.19 nM T98691 C5M1BT 25195691 IC50 = 3162.28 nM T98691 CC7TV3 25204336 IC50 > 10000 nM T98691 C73KLE 25209862 IC50 = 4.67 nM T98691 C9FWJ4 25219913 IC50 = 32850 nM T98691 CJ04ZN 25234563 IC50 = 152 nM T98691 CU59SO 25242431 Ki = 16000 nM T98691 C23JPC 25242432 Ki = 14000 nM T98691 CW9JM2 25256832 IC50 = 2000 nM T98691 C3GC7P 25256833 IC50 = 1400 nM T98691 CXU0P9 26794600 Ki = 64000 nM T98691 CTME03 38864605 IC50 = 3150 nM T98691 C26LPI 38864607 IC50 = 9420 nM T98691 CN80BC 38864634 IC50 = 56510 nM T98691 CE4D9Q 40522013 Ki = 17000 nM T98691 CL96WQ 42633150 IC50 = 5246 nM T98691 CZ5F4C 42633340 IC50 = 711 nM T98691 C5XV0H 42633341 IC50 = 49 nM T98691 CZS24P 42633520 IC50 = 98 nM T98691 CI78XT 42633521 IC50 = 1060 nM T98691 CU6PL7 42633691 IC50 = 1086 nM T98691 CQ9TR8 42633692 IC50 = 966 nM T98691 C6FJW2 42634249 IC50 = 1084 nM T98691 C9EN0G 42634411 IC50 = 426 nM T98691 C2ZXJ7 42634578 IC50 = 631 nM T98691 CI25RJ 42634754 IC50 = 436 nM T98691 CZ6B1F 42635119 IC50 = 121 nM T98691 C5X4WG 42635483 IC50 = 219 nM T98691 CZM36T 42641892 IC50 > 10000 nM T98691 CRYH80 42642459 IC50 > 10000 nM T98691 C3DC4M 42647278 Ki = 0.87 nM T98691 C25ELB 44143088 IC50 = 117.49 nM T98691 CL0M7R 44143089 IC50 = 7943.28 nM T98691 C9QDC0 44143091 IC50 = 562.34 nM T98691 CNM6X8 44218399 IC50 = 625 nM T98691 C8Y9NQ 44219712 IC50 = 1240 nM T98691 CJA68L 44224113 IC50 = 251.19 nM T98691 C2V5ZT 44224114 IC50 = 1258.93 nM T98691 C0U9VJ 44224115 IC50 = 501.19 nM T98691 C0MZ9D 44224116 IC50 = 316.23 nM T98691 CEJ82A 44224117 IC50 = 251.19 nM T98691 C0KL7D 44224118 IC50 = 251.19 nM T98691 CE9S0M 44224119 IC50 = 794.33 nM T98691 CV1W0Z 44224120 IC50 = 79.43 nM T98691 C5LDK7 44224121 IC50 = 79.43 nM T98691 C8UF5Q 44224122 IC50 = 316.23 nM T98691 C9YHC5 44224123 IC50 = 50.12 nM T98691 CA26RI 44224124 IC50 = 251.19 nM T98691 CU0PI2 44224125 IC50 = 398.11 nM T98691 CRL79W 44224126 IC50 = 100 nM T98691 C3T0QO 44224127 IC50 = 19.95 nM T98691 C81EVM 44224128 IC50 = 1258.93 nM T98691 C7IY8P 44224129 IC50 = 501.19 nM T98691 CYG02V 44224130 IC50 = 630.96 nM T98691 CJS1B9 44224131 IC50 = 398.11 nM T98691 CN5O8S 44224132 IC50 = 79.43 nM T98691 C2Q3RP 44224133 IC50 = 63.1 nM T98691 CZX62T 44224134 IC50 = 79.43 nM T98691 CP3YA9 44224135 IC50 = 12.59 nM T98691 CSZH31 44224136 IC50 = 12.59 nM T98691 CZ56BP 44263398 IC50 > 20000 nM T98691 CR38EU 44279051 Ki = 47 nM T98691 C5LJS7 44279083 Ki = 16 nM T98691 C2V7RL 44279437 Ki = 39 nM T98691 CD84XF 44279475 IC50 = 15 nM T98691 C0RQ3V 44279712 IC50 = 2.6 nM T98691 CFJ2Z1 44279771 IC50 = 17 nM T98691 C3IBQ0 44279792 IC50 = 3960 nM T98691 CQ57HR 44279823 IC50 = 163 nM T98691 C5YF0J 44279873 IC50 = 37400 nM T98691 C6ZXK0 44280152 IC50 = 166 nM T98691 CVZ54E 44280172 IC50 = 47 nM T98691 CCPA17 44294490 Ki = 90 nM T98691 C2ZHC1 44295739 IC50 = 5400 nM T98691 CNL8Y4 44302956 IC50 = 130 nM T98691 CAM2S5 44302974 IC50 > 10000 nM T98691 CBYD40 44302975 IC50 = 580 nM T98691 CNA24Z 44303031 IC50 > 10000 nM T98691 C56IEO 44303058 IC50 = 10000 nM T98691 CL4VM1 44303061 IC50 > 10000 nM T98691 CS0P5A 44303274 IC50 > 10000 nM T98691 CXU16T 44303285 IC50 = 6000 nM T98691 CEIH70 44303290 IC50 > 10000 nM T98691 CN21AS 44303309 IC50 > 10000 nM T98691 C24EDH 44303315 IC50 = 10000 nM T98691 CDX5M7 44303318 IC50 = 6900 nM T98691 CRK48P 44303319 IC50 > 10000 nM T98691 CKB9O1 44303324 IC50 = 1300 nM T98691 C0FEJ1 44303335 IC50 < 30 nM T98691 CT49MJ 44303338 IC50 = 150 nM T98691 CMF6W2 44303344 IC50 = 30 nM T98691 CD1HJ5 44303345 IC50 = 580 nM T98691 CL26OE 44303389 IC50 = 90 nM T98691 CN9QY5 44303414 IC50 = 10000 nM T98691 CG3OM8 44304535 Ki = 3400 nM T98691 C0FKB3 44304563 Ki = 140000 nM T98691 CC04TQ 44304591 Ki > 150000 nM T98691 C76OIY 44304610 Ki = 3700 nM T98691 CK8JW5 44304611 Ki > 150000 nM T98691 CZ87NW 44304634 Ki > 150000 nM T98691 COR96D 44304861 Ki = 16000 nM T98691 C9O1VP 44319528 Ki = 12 nM T98691 CH9E6N 44321598 Ki = 30 nM T98691 C6EYQ8 44321883 Ki = 29 nM T98691 CTW41Y 44321884 Ki = 52 nM T98691 CU7J2P 44321946 Ki = 154 nM T98691 CKB02C 44329582 Ki = 6340 nM T98691 CTN34G 44329585 Ki = 130 nM T98691 CR1J6F 44329593 Ki = 3000 nM T98691 C3EHF1 44329596 Ki = 790 nM T98691 C97WPV 44329608 Ki = 760 nM T98691 CY5KH4 44329643 Ki = 16700 nM T98691 CJ5W0G 44332538 Ki = 597 nM T98691 C1KD2V 44332539 Ki = 865 nM T98691 C7XQY2 44332540 Ki = 93 nM T98691 C2FHG7 44332555 Ki = 377 nM T98691 C6QOU0 44332714 Ki = 232 nM T98691 C83QDU 44332915 Ki = 299.4 nM T98691 CNO3T1 44342482 IC50 = 0.74 nM T98691 C1IJW5 44343023 IC50 = 8500 nM T98691 C71JRX 44343028 IC50 = 15 nM T98691 COEK09 44343037 IC50 = 270 nM T98691 C61UIS 44343092 IC50 = 110 nM T98691 CB64RL 44343105 IC50 = 1200 nM T98691 C0TAX2 44345292 Ki = 55 nM T98691 CD9P4K 44345387 Ki > 1000 nM T98691 C8HP5M 44347822 IC50 = 2163 nM T98691 CK0B9C 44347827 IC50 > 10000 nM T98691 CO82ZV 44347993 IC50 > 10000 nM T98691 CLCP51 44348116 IC50 = 919 nM T98691 CFBI42 44348134 IC50 = 5783 nM T98691 CYEI89 44348185 IC50 = 338 nM T98691 C3V0GM 44348957 IC50 > 1000 nM T98691 CFI6N5 44348963 IC50 = 23 nM T98691 CNZ2I9 44353889 IC50 = 2400 nM T98691 C9EOS5 44353924 IC50 > 1000 nM T98691 CG1JP8 44353951 IC50 = 1100 nM T98691 CX1IL0 44353974 IC50 = 220 nM T98691 CQ1F6V 44353976 IC50 = 560 nM T98691 CJA79K 44353977 IC50 > 1000 nM T98691 C3GV4U 44353978 IC50 = 1400 nM T98691 C67ZFU 44353986 IC50 = 2800 nM T98691 CT7JK8 44354015 IC50 = 210 nM T98691 C49VSE 44354016 IC50 = 6100 nM T98691 CAC2Q0 44356377 IC50 = 1.4 nM T98691 CU6KO2 44356379 IC50 = 150 nM T98691 C6JTS1 44356381 IC50 = 4.3 nM T98691 CYK6F4 44356399 IC50 = 0.95 nM T98691 CUJK15 44356612 IC50 = 0.74 nM T98691 CBPJ08 44356625 IC50 = 95 nM T98691 C0DE5P 44356626 IC50 = 0.95 nM T98691 CI9OQ6 44356637 IC50 = 3.1 nM T98691 CRA87Z 44356780 IC50 = 4.5 nM T98691 CH9L1E 44356846 IC50 = 5.3 nM T98691 CKS7I4 44357044 IC50 = 0.97 nM T98691 C35ROP 44357071 IC50 = 2.2 nM T98691 C7DOS2 44366435 Ki > 100000 nM T98691 CA9LC3 44382185 Ki = 9 nM T98691 C5NH3W 44382186 Ki = 1 nM T98691 CZU70X 44382187 Ki = 1 nM T98691 C3M5CT 44382237 Ki = 36 nM T98691 C3W7CI 44382238 Ki = 1 nM T98691 CM9WG5 44382239 Ki = 32 nM T98691 CUEX04 44382949 Ki = 7844 nM T98691 C9UQN0 44383254 Ki > 10000 nM T98691 CU4CB8 44383255 Ki = 4110 nM T98691 C83ART 44383306 Ki = 2 nM T98691 CEUA60 44383413 Ki = 2 nM T98691 CX20UA 44383464 Ki = 230 nM T98691 CP7KW2 44391459 IC50 = 130 nM T98691 C9W3HN 44391474 IC50 = 0.71 nM T98691 CV71WQ 44391475 IC50 = 81 nM T98691 CIG5R6 44393795 IC50 = 458 nM T98691 C78QJO 44394249 Ki = 107000 nM T98691 CQRB69 44394250 Ki = 51000 nM T98691 CTRP74 44394287 IC50 = 3000 nM T98691 CP7X6J 44394353 IC50 = 1200 nM T98691 C79NFU 44394458 IC50 = 3000 nM T98691 C2J6MW 44397423 IC50 = 15000 nM T98691 CRSF50 44397609 IC50 = 37000 nM T98691 CHWX97 44397693 IC50 = 130000 nM T98691 CZC50Y 44398247 IC50 > 10000 nM T98691 CQPM06 44398248 IC50 > 10000 nM T98691 CYJ8Z4 44398353 IC50 = 430 nM T98691 CD73QR 44398649 Ki = 0.79 nM T98691 CHQF16 44398651 Ki = 0.025 nM T98691 C4ALQ9 44398659 Ki = 1500 nM T98691 CGQ20I 44398741 Ki = 0.036 nM T98691 CD18YP 44402055 IC50 = 660 nM T98691 CU8TB9 44402056 IC50 = 2600 nM T98691 CD4TP7 44402158 IC50 = 460 nM T98691 CO6BG2 44402160 IC50 = 1700 nM T98691 C0AJC4 44402175 IC50 = 6800 nM T98691 CX9O2Q 44402263 IC50 = 4400 nM T98691 C89MOT 44402291 IC50 = 1000 nM T98691 CFL9B8 44402952 IC50 = 68 nM T98691 CRZT97 44403028 IC50 > 10000 nM T98691 CW2L5D 44404573 Ki = 673 nM T98691 C39PTS 44404574 Ki = 251 nM T98691 CY5NW9 44405210 Ki = 4000 nM T98691 CP8L2A 44405213 Ki = 7500 nM T98691 CA59MJ 44405279 Ki = 22000 nM T98691 C5GS4Y 44405280 Ki > 150000 nM T98691 CDP93F 44405305 Ki = 14000 nM T98691 C64UAX 44405607 Ki = 6400 nM T98691 CI9P8B 44405608 Ki = 4800 nM T98691 C4ZMP9 44408016 IC50 = 11000 nM T98691 C25RIN 44408049 IC50 = 12 nM T98691 C9IEW7 44409018 Ki = 1754 nM T98691 CKC4P5 44411027 Ki = 6000 nM T98691 C2MDN7 44411237 Ki = 4000 nM T98691 CY4H2I 44411981 Ki = 1300 nM T98691 CNU4T9 44412155 Ki = 1 nM T98691 CYF1B9 44412339 Ki > 150000 nM T98691 C1J6OW 44412340 Ki > 150000 nM T98691 CU49OM 44412341 Ki = 63000 nM T98691 CDK32G 44412349 Ki = 4600 nM T98691 CL82XD 44412354 Ki = 100000 nM T98691 C23ZVR 44412355 Ki = 28000 nM T98691 CV26BC 44412365 Ki = 14000 nM T98691 CX93NW 44412366 Ki = 2100 nM T98691 CZN9T0 44412387 Ki = 160 nM T98691 CY90QW 44412402 Ki = 2900 nM T98691 C1HW8F 44412424 Ki = 2900 nM T98691 CYDJ14 44412436 Ki = 960 nM T98691 CV49GB 44412437 Ki = 150000 nM T98691 CZ5VW2 44412440 Ki = 18000 nM T98691 CZR1O3 44412502 Ki = 130000 nM T98691 CA23SL 44414977 Ki = 2500 nM T98691 C0XB2M 44414978 Ki = 360 nM T98691 CAG5F3 44414992 Ki = 680 nM T98691 C8JL9C 44415006 Ki = 540 nM T98691 CS6X7V 44426055 IC50 = 994 nM T98691 C8IB2W 44426056 IC50 > 100000 nM T98691 CVD7L4 44442257 IC50 = 3389 nM T98691 C3J4DH 44444205 IC50 = 96 nM T98691 CX15UA 44444919 IC50 = 2380 nM T98691 CUXF67 44444920 IC50 = 5830 nM T98691 C1DHA5 44444921 IC50 = 9400 nM T98691 CJWB56 44444922 IC50 = 11780 nM T98691 C0NB8D 44444923 IC50 > 30000 nM T98691 C9P7OQ 44444924 IC50 = 870 nM T98691 CXO56L 44447657 IC50 = 2940 nM T98691 CB6H5U 44447658 IC50 > 10000 nM T98691 C1U6JA 44447659 IC50 = 456 nM T98691 CV3T1A 44447660 IC50 > 10000 nM T98691 CF7AV1 44447661 IC50 = 262 nM T98691 C7HRP2 44447662 IC50 = 2650 nM T98691 C0CZ7P 44447663 IC50 = 472 nM T98691 CAF54M 44447664 IC50 = 110 nM T98691 CC4J7S 44447665 IC50 = 750 nM T98691 C7QW0F 44449893 IC50 = 118 nM T98691 CW30VS 44449926 IC50 = 21 nM T98691 C40EDY 44449928 IC50 = 44 nM T98691 C83KAR 44449929 IC50 = 39 nM T98691 C59IFW 44449957 IC50 = 17 nM T98691 CH7YE8 44449958 IC50 = 11 nM T98691 CTQ3A1 44449959 IC50 = 81 nM T98691 CF59ZH 44449960 IC50 = 7.4 nM T98691 C59OXW 44449989 IC50 = 9.4 nM T98691 C69NRS 44449990 IC50 = 3.6 nM T98691 C3KV1I 44450083 IC50 = 2998 nM T98691 CB38OA 44450114 IC50 = 110 nM T98691 C5RQF1 44450115 IC50 = 201 nM T98691 CZU1L6 44450142 IC50 = 21797 nM T98691 CQ7S0A 44450143 IC50 = 41 nM T98691 CNJ3P7 44450179 IC50 = 115 nM T98691 CL6WZ1 44450271 IC50 = 980 nM T98691 C3B2TR 44450349 IC50 > 1000 nM T98691 C38JBH 44450361 IC50 > 1000 nM T98691 CC0AG3 44452909 Ki = 220 nM T98691 CB8IX2 44452912 Ki = 70 nM T98691 CXJF30 44452936 Ki = 30 nM T98691 CVCJ36 44452938 Ki = 1 nM T98691 C4ZBF6 44452963 Ki = 28000 nM T98691 CWCK10 44452964 Ki = 14000 nM T98691 CF9PC3 44452965 Ki = 100000 nM T98691 CF57UN 44456198 IC50 = 133 nM T98691 CKNS35 44456237 IC50 = 34000 nM T98691 C5I2XF 44457308 Ki = 14000 nM T98691 C7HM2X 44457465 Ki = 10700 nM T98691 C91IOW 44457476 Ki = 6000 nM T98691 C2G7LZ 44457481 Ki = 511 nM T98691 C5I0JY 44457489 Ki = 464 nM T98691 CM14NI 44457496 Ki = 24 nM T98691 C70HBQ 44457499 Ki = 21 nM T98691 COR85M 44457502 Ki = 23 nM T98691 C0O8XF 44457507 Ki = 112 nM T98691 CX49LO 44457510 Ki = 45 nM T98691 CKV1E8 44457511 Ki = 155 nM T98691 CIT48F 44457512 Ki = 460 nM T98691 CTUD83 44457513 Ki = 19 nM T98691 C0B4IO 44457516 Ki = 57500 nM T98691 C8Z4WO 44459967 IC50 = 309.03 nM T98691 C86ORE 44459987 IC50 = 204.17 nM T98691 C9TFJ8 44464926 IC50 = 1258.93 nM T98691 CYO0T1 44465454 IC50 = 39.81 nM T98691 CE83YL 44465721 IC50 = 25.12 nM T98691 CVD48M 44478848 IC50 = 730 nM T98691 CJR45G 44479122 IC50 = 355 nM T98691 C8I9QK 44479381 IC50 = 610 nM T98691 CWS3K7 44479385 IC50 = 240 nM T98691 C2PK4G 44479635 IC50 = 48 nM T98691 CB73NC 44479637 IC50 = 145 nM T98691 CA48JP 44480468 IC50 = 1400 nM T98691 C0ZE3C 44480469 IC50 = 1500 nM T98691 C0G5ET 44480470 IC50 = 700 nM T98691 CH7I8C 44480471 IC50 = 400 nM T98691 CPDQ74 44480723 IC50 = 1900 nM T98691 CPN9C7 44480724 IC50 = 1100 nM T98691 CZ62AB 44480725 IC50 = 900 nM T98691 C8SL0N 44480726 IC50 = 2700 nM T98691 C1ZOM7 44480727 IC50 = 900 nM T98691 CZE95Q 44480728 IC50 = 480 nM T98691 CYBH29 44480974 IC50 = 6000 nM T98691 CA0F2M 44480975 IC50 = 460 nM T98691 CFJ21O 44480976 IC50 = 16000 nM T98691 C94NWI 44480977 IC50 = 1000 nM T98691 CFE2H6 44480978 IC50 = 800 nM T98691 COJ38W 44480979 IC50 = 1500 nM T98691 C45EMI 44481231 IC50 = 800 nM T98691 COL4C2 44481232 IC50 = 1400 nM T98691 CJ1M6E 44481233 IC50 = 1100 nM T98691 C32YDM 44481234 IC50 = 1800 nM T98691 CG1X4W 44481235 IC50 = 1600 nM T98691 CG5YU6 44481236 IC50 = 1300 nM T98691 CUHM64 44481503 IC50 = 800 nM T98691 CBGO51 44481504 IC50 = 840 nM T98691 CT9W2X 44481505 IC50 = 600 nM T98691 C1S0KC 44481506 IC50 = 1600 nM T98691 CRQ32O 44481507 IC50 = 190 nM T98691 C1E6AT 44481508 IC50 = 1800 nM T98691 CCW6N4 44481776 IC50 = 1000 nM T98691 CCOK78 44481777 IC50 = 1100 nM T98691 CK1E7H 44481778 IC50 = 900 nM T98691 CFYP92 44482496 IC50 = 130 nM T98691 C1LWX5 44552274 Ki = 4200 nM T98691 CIP6M8 44552275 Ki = 4100 nM T98691 C8W2LG 44552367 Ki = 39700 nM T98691 CWJV95 44552368 Ki = 7700 nM T98691 CIT5G7 44561891 IC50 > 100000 nM T98691 C90BGR 44561892 IC50 > 100000 nM T98691 C9RGX4 44561893 IC50 > 100000 nM T98691 CU7NP5 44561930 IC50 > 100000 nM T98691 CV21IQ 44561931 IC50 > 100000 nM T98691 CR08WA 44561932 IC50 > 100000 nM T98691 CV1IL5 44565796 IC50 > 10000 nM T98691 CLH74F 44565900 IC50 = 1060 nM T98691 CMIP10 44565901 IC50 = 1000 nM T98691 C70BXJ 44565925 IC50 = 1370 nM T98691 CS6YO0 44566187 IC50 = 0.437 nM T98691 CSF17Z 44566188 IC50 > 100000 nM T98691 CJP3U5 44566195 IC50 = 1.66 nM T98691 CUFJ57 44566196 IC50 = 19820 nM T98691 CI6H7R 44568190 IC50 > 2000 nM T98691 CVX81T 44568191 IC50 > 5000 nM T98691 CJRQ74 44568192 IC50 > 1000 nM T98691 C6ZHA4 44568193 IC50 > 1000 nM T98691 C2X3HJ 44568223 IC50 > 1000 nM T98691 CV54EU 44568306 IC50 > 4000 nM T98691 CDZ03Q 44568307 IC50 > 1000 nM T98691 C6FV7W 44568638 IC50 > 1000 nM T98691 C6U3RB 44568639 IC50 = 370 nM T98691 COJ16S 44568640 IC50 = 320 nM T98691 CVP4Y6 44568641 IC50 > 1000 nM T98691 CZW5K2 44568669 IC50 = 260 nM T98691 CW89JM 44568670 IC50 = 840 nM T98691 C2D9TS 44568671 IC50 > 1000 nM T98691 CU4PO0 44568672 IC50 = 23 nM T98691 CCJ68F 44568673 IC50 = 86 nM T98691 CCIP49 44568714 IC50 = 40 nM T98691 C3HYW8 44568715 IC50 > 1000 nM T98691 CLXN21 44568716 IC50 > 1000 nM T98691 CA86UV 44568718 IC50 > 1000 nM T98691 CU82VX 44568766 IC50 > 1000 nM T98691 CZF5G0 44568767 IC50 > 1000 nM T98691 CVR02S 44568768 IC50 > 1000 nM T98691 C1P3LN 44568769 IC50 = 790 nM T98691 CG74ZL 44568770 IC50 > 1000 nM T98691 COHB20 44570671 Ki = 12000 nM T98691 C35ZYP 44570672 Ki = 64000 nM T98691 C3BHM4 44570673 Ki = 16000 nM T98691 C0OSY2 44570674 Ki = 11000 nM T98691 CF41YI 44570719 Ki = 15000 nM T98691 CY9ZT4 44570833 Ki = 7200 nM T98691 CB3S2D 44570834 Ki = 29000 nM T98691 C8K6PB 44570835 Ki = 2000 nM T98691 CWH9Q0 44570836 Ki = 23000 nM T98691 CA10KC 44570876 Ki = 970 nM T98691 CAUD26 44570877 Ki = 7800 nM T98691 C1XCP6 44570878 Ki = 9500 nM T98691 CN1GT2 44570879 Ki = 2300 nM T98691 CV0KJ4 44570915 Ki = 1100 nM T98691 C14JNH 44570916 Ki = 31000 nM T98691 C1DA8K 44570917 Ki = 14000 nM T98691 C9CMZ2 44570957 Ki = 5900 nM T98691 C37LRT 44570958 Ki = 7800 nM T98691 C31BXW 44570959 Ki = 11000 nM T98691 C5G2KT 44570997 Ki = 8400 nM T98691 CZ1ET3 44570998 Ki = 9100 nM T98691 CSYI14 44570999 Ki = 11000 nM T98691 CK5ZM6 44571085 Ki = 7900 nM T98691 CNP2G3 44571086 Ki = 6800 nM T98691 CX2B3F 44571130 Ki = 8500 nM T98691 CFTE86 44571131 Ki = 13000 nM T98691 C4DV1E 44571132 Ki = 14000 nM T98691 C05LYD 44571173 Ki = 13000 nM T98691 CC5A6D 44571174 Ki = 8700 nM T98691 CHB7Y3 44571175 Ki = 23000 nM T98691 C6XF8B 44571212 Ki = 13000 nM T98691 CG5ZO3 44571213 Ki = 24000 nM T98691 C67UMF 44571214 Ki = 27000 nM T98691 CD6X2Y 44571254 Ki = 9100 nM T98691 CQ0W5J 44571255 Ki = 17000 nM T98691 CGM30J 44571297 Ki = 10000 nM T98691 CU0D3P 44571298 Ki = 12000 nM T98691 CUG72S 44571323 Ki = 2500 nM T98691 C2NT4H 44571324 Ki = 11000 nM T98691 CC12QS 44571325 Ki = 27000 nM T98691 CI39YN 44571326 Ki = 15000 nM T98691 C1L3KX 44571358 Ki = 17000 nM T98691 C0NFJ8 44571359 Ki = 21000 nM T98691 CE2PQ4 44571360 Ki = 15000 nM T98691 C5S6FJ 44571361 Ki = 15000 nM T98691 C8YPA6 44572419 Ki = 7400 nM T98691 C3L7IV 44572420 Ki = 2700 nM T98691 CFZ3L7 44572422 Ki = 1900 nM T98691 CFZB79 44572423 Ki = 8400 nM T98691 CGC0W5 44572424 Ki = 3200 nM T98691 C9E6QP 44579079 IC50 = 426 nM T98691 C7CKG9 44579080 IC50 = 276 nM T98691 CFN0Z1 44579081 IC50 > 1000 nM T98691 CH5B0N 44579120 IC50 = 440 nM T98691 CN42GY 44579121 IC50 = 360 nM T98691 CDUJ10 44579122 IC50 = 400 nM T98691 CQJ0L6 44579123 IC50 = 330 nM T98691 CO13BP 44579170 IC50 = 300 nM T98691 CP0X4D 44579171 IC50 = 460 nM T98691 CS60PG 44579172 IC50 = 1390 nM T98691 CY2E6M 44579173 IC50 = 2500 nM T98691 CA0OT2 44587365 IC50 = 64 nM T98691 CM35BH 44587366 IC50 = 270 nM T98691 C2AVQ0 44587440 IC50 = 870 nM T98691 CO7TR5 44587827 IC50 > 2000 nM T98691 CL18MT 44587828 IC50 = 2000 nM T98691 C3A4JO 44587829 IC50 = 780 nM T98691 C9HES8 44587858 IC50 > 3000 nM T98691 CA4DK2 44587859 IC50 > 3000 nM T98691 C76PSY 44587860 IC50 > 3000 nM T98691 C6NU0J 44587861 IC50 > 3000 nM T98691 C8C1OM 44587862 IC50 = 840 nM T98691 CERA06 44587897 IC50 = 1500 nM T98691 CI87JG 44587898 IC50 = 480 nM T98691 C2OQE5 44587899 IC50 = 840 nM T98691 CNM2G4 44587937 IC50 = 700 nM T98691 C65NLR 44587938 IC50 = 510 nM T98691 C81ZSB 44587939 IC50 = 100 nM T98691 CX40GW 46226591 Ki = 850 nM T98691 C8HEC4 46226622 Ki = 13600 nM T98691 CELQ42 46226646 Ki = 7000 nM T98691 CA7V4F 46226655 Ki = 2100 nM T98691 C4YAJ7 46228924 IC50 > 10000000 nM T98691 CD1W6B 46232382 IC50 > 10000 nM T98691 CRYZ16 46232383 IC50 > 10000 nM T98691 C60TNV 46232384 IC50 > 10000 nM T98691 C1I8LN 46232385 IC50 = 2460 nM T98691 C4P7CD 46232387 IC50 > 10000 nM T98691 CQN2I7 46232805 IC50 = 30.5 nM T98691 C39QNG 46232806 IC50 = 1610 nM T98691 CFW92U 46232807 IC50 = 2600 nM T98691 CWD0B5 46232808 IC50 > 10000 nM T98691 CPB62W 46232809 IC50 = 250 nM T98691 CU8ZB6 46232845 IC50 = 131 nM T98691 C32ENI 46232846 IC50 = 46.5 nM T98691 CX0O3T 46232848 IC50 = 79.6 nM T98691 C0WJ4R 46232849 IC50 = 327 nM T98691 CU5KA6 46232850 IC50 > 10000 nM T98691 C5W2SX 46232966 IC50 = 521 nM T98691 CEJ0Z8 46232968 IC50 = 83.8 nM T98691 C60SCN 46232969 IC50 = 610 nM T98691 CL6GY7 46232970 IC50 = 59.4 nM T98691 CA9QH7 46232971 IC50 = 415 nM T98691 C8N2YC 46233007 IC50 = 96 nM T98691 C8HR1S 46233008 IC50 = 233 nM T98691 CY84AW 46233009 IC50 = 114 nM T98691 CRS52G 46233010 IC50 = 118 nM T98691 CC64UL 46233011 IC50 = 63.2 nM T98691 C0U9OQ 46233012 IC50 > 10000 nM T98691 CV74LQ 46233041 IC50 = 2220 nM T98691 C1ZG2T 46233042 IC50 > 10000 nM T98691 C6IJO8 46233043 IC50 = 3320 nM T98691 CZ1E0U 46233044 IC50 > 10000 nM T98691 CH29YW 46233045 IC50 > 10000 nM T98691 CO94IL 46233046 IC50 > 10000 nM T98691 COEI67 46233047 IC50 = 4570 nM T98691 CC2N0F 46842579 IC50 > 10000 nM T98691 CV6SW4 46842581 IC50 > 10000 nM T98691 CM2D1G 46842582 IC50 > 10000 nM T98691 CIU1R5 46842626 IC50 > 10000 nM T98691 C37OSC 46842709 IC50 > 10000 nM T98691 C6HD4M 46865101 IC50 > 10000 nM T98691 CC7DG3 46866398 IC50 = 9772 nM T98691 CGT1Z2 46881448 IC50 > 10000 nM T98691 CH9ON3 46881449 IC50 > 10000 nM T98691 CF15KQ 46881450 IC50 > 10000 nM T98691 CN58BG 46882092 IC50 > 10000 nM T98691 CG9X3C 46882094 IC50 > 10000 nM T98691 CZ5KP8 46882095 IC50 > 10000 nM T98691 CPQZ83 46882096 IC50 > 10000 nM T98691 CUI91D 46905615 IC50 = 560 nM T98691 CS4VM8 46945615 IC50 = 22 nM T98691 CFWU08 46946224 IC50 > 25000 nM T98691 CVT40A 46947220 IC50 = 29700 nM T98691 CAFW31 49783666 IC50 > 10000 nM T98691 CJH50R 49797481 IC50 > 100000 nM T98691 CI7P2B 49797571 IC50 = 15500 nM T98691 CI59MV 49797572 IC50 > 50000 nM T98691 C96CKU 49797573 IC50 = 5400 nM T98691 C9LNK5 49798881 Ki > 150000 nM T98691 CE6Z7V 49798882 Ki = 59900 nM T98691 C5CY7U 49798883 Ki = 12000 nM T98691 C3B8FE 49798886 Ki = 12200 nM T98691 C8R6CQ 49798901 Ki = 2700 nM T98691 C7YZV2 49798902 Ki = 76500 nM T98691 CO7I0B 49798903 Ki = 65000 nM T98691 CVT4U3 49798904 Ki > 150000 nM T98691 C3Y6OC 49798905 Ki = 29800 nM T98691 C4NB3R 49834903 IC50 = 4200 nM T98691 CQ3W9J 49834904 IC50 = 4600 nM T98691 CX1WU8 49834905 IC50 = 2600 nM T98691 CA96LF 49834906 IC50 = 16200 nM T98691 CB9MS2 49834907 IC50 = 2700 nM T98691 C74RAF 49834908 IC50 = 4100 nM T98691 CN8E2A 49834971 IC50 = 1900 nM T98691 COG9T6 49834972 IC50 = 15800 nM T98691 CGPM91 49834975 IC50 = 17000 nM T98691 CJ73DH 49835032 IC50 = 33600 nM T98691 C8XR4Q 49835033 IC50 = 4700 nM T98691 CXE51M 49835035 IC50 = 24900 nM T98691 CKRG17 49835144 IC50 > 25000 nM T98691 C9NO4U 49835145 IC50 > 25000 nM T98691 CP4S5A 49835673 IC50 = 11700 nM T98691 CS3HC6 49835674 IC50 = 12200 nM T98691 C8O3UF 49835732 IC50 = 22200 nM T98691 C37RZT 49862146 IC50 > 10000 nM T98691 CJ0HY8 49862186 IC50 > 10000 nM T98691 CKA53W 49862308 IC50 > 10000 nM T98691 C8B2WE 49862309 IC50 > 10000 nM T98691 CR13LF 49862310 IC50 > 10000 nM T98691 C38BJK 49862365 IC50 > 10000 nM T98691 C1Z9VQ 49862366 IC50 > 10000 nM T98691 C6W1UJ 49862367 IC50 > 10000 nM T98691 CIFP19 49862368 IC50 > 10000 nM T98691 CMW23V 49862369 IC50 > 10000 nM T98691 CI4J0A 49862370 IC50 > 10000 nM T98691 C1XBM6 49862420 IC50 > 10000 nM T98691 CKV06S 49862421 IC50 > 10000 nM T98691 CN4GD6 49862422 IC50 > 10000 nM T98691 CA7K8Q 49862423 IC50 > 10000 nM T98691 CS92IZ 49862471 IC50 > 10000 nM T98691 C1NAQ5 49862472 IC50 > 10000 nM T98691 C5OD6J 49862473 IC50 > 10000 nM T98691 CFCH31 49862474 IC50 > 10000 nM T98691 C29OGE 49862475 IC50 > 10000 nM T98691 CVOG15 49865938 Ki > 100000 nM T98691 CRI85M 50898446 IC50 = 150.8 nM T98691 C18RNG 50925386 Ki = 2700 nM T98691 C4I0JY 50925524 IC50 = 42 nM T98691 C01DJG 50993971 Ki = 860 nM T98691 CW9X3R 50993972 Ki = 480 nM T98691 CIC7H1 50993973 Ki = 1.5 nM T98691 C3UB9Y 50993974 Ki = 2.6 nM T98691 CMS13V 50994055 Ki = 0.4 nM T98691 CPT6I5 50994056 Ki = 0.36 nM T98691 CB4X6Y 50994057 Ki = 0.045 nM T98691 CSY4W0 50994058 Ki = 0.39 nM T98691 CQ08HC 50994059 Ki = 1.4 nM T98691 C30WKN 50994060 Ki = 1.1 nM T98691 C8A1GN 50994137 Ki = 2 nM T98691 C6K3EJ 50994138 Ki = 4.4 nM T98691 CN6ZM0 50994139 Ki = 4700 nM T98691 CF7SN9 50994140 Ki = 940 nM T98691 CU7M1P 50994141 Ki > 22000 nM T98691 C4FE0T 50994142 Ki = 0.22 nM T98691 CJ86MG 51031171 IC50 = 30 nM T98691 C8I1YU 51031462 IC50 = 12 nM T98691 CI1H9F 51031463 IC50 = 6.5 nM T98691 CKNC78 51031601 IC50 = 6.5 nM T98691 CS9Z0X 51031602 IC50 = 4.3 nM T98691 C96FHG 51033722 IC50 = 3600 nM T98691 C6JU9I 51347016 Ki = 690 nM T98691 C2C1YQ 51347017 Ki = 33 nM T98691 C4JB5S 52941092 IC50 > 10000 nM T98691 CDC64G 52941172 IC50 > 10000 nM T98691 C7DO0F 52941283 IC50 = 751 nM T98691 CU1TW6 52941414 IC50 = 458 nM T98691 C71VFU 52941469 IC50 = 891 nM T98691 C8BP5L 52941833 IC50 = 814.5 nM T98691 CQ39TK 52941839 IC50 = 931.3 nM T98691 CDO45C 52941841 IC50 > 10000 nM T98691 CW05MV 52942797 IC50 = 141 nM T98691 C9MK7J 52942931 IC50 = 3819 nM T98691 CVO3U2 52943063 IC50 > 10000 nM T98691 C2AV9H 52943244 IC50 > 10000 nM T98691 CYLF86 52943307 IC50 > 10000 nM T98691 CQDG96 52943578 IC50 > 10000 nM T98691 C4TY6S 52943722 IC50 > 10000 nM T98691 CQ6N0I 52943841 IC50 > 10000 nM T98691 C9B6DJ 52944285 Ki = 3.7 nM T98691 C1UP6N 52945298 IC50 > 10000 nM T98691 CF1LS6 52945475 IC50 > 10000 nM T98691 CN6V0H 52945759 IC50 = 9650 nM T98691 CV8L9Z 52945985 IC50 = 379 nM T98691 CLJ83U 52946267 IC50 > 10000 nM T98691 CBD6S0 52946687 IC50 = 369.7 nM T98691 CS2NX6 52946690 IC50 > 10000 nM T98691 CND9C6 52947170 IC50 > 10000 nM T98691 CT28XU 52947761 IC50 = 2628 nM T98691 CI0S1W 52947952 IC50 > 10000 nM T98691 C75SHQ 52948860 IC50 = 479 nM T98691 C56OCA 53317528 IC50 = 630.96 nM T98691 CM60RJ 53317530 IC50 = 12589.25 nM T98691 C5A6IH 53317737 IC50 = 1258.93 nM T98691 C6FEH9 53318816 IC50 > 25118.86 nM T98691 CJAX07 53318817 IC50 = 2511.89 nM T98691 CG5AP6 53318818 IC50 = 3162.28 nM T98691 CJ3PN0 53319501 IC50 > 10000 nM T98691 C7V2DA 53322116 IC50 > 10000 nM T98691 CQ8O1R 53322117 IC50 > 10000 nM T98691 CR1L4Y 53325394 IC50 > 25118.86 nM T98691 CWJB05 53364091 IC50 = 429 nM T98691 CPN6B8 53378493 IC50 = 9000 nM T98691 C1NJ6T 56654510 Ki > 5000 nM T98691 CDAN29 56657787 IC50 = 3.3 nM T98691 CU26MD 56657788 IC50 = 3.9 nM T98691 CD5W7V 56661312 IC50 = 2 nM T98691 CIX1H6 56664780 IC50 = 6.1 nM T98691 C24ZAM 56664781 IC50 = 2 nM T98691 C24PVH 56664782 IC50 = 3.3 nM T98691 C70CMI 56664783 IC50 = 7.1 nM T98691 CCG3S4 56666730 IC50 = 10 nM T98691 CB57PR 56668196 IC50 = 2.2 nM T98691 CK54CF 56670150 IC50 = 0.53 nM T98691 C69ILG 56670151 IC50 = 22.4 nM T98691 CU59KM 56671669 IC50 = 4.5 nM T98691 C46EFG 56675090 IC50 = 2.1 nM T98691 CDN7E0 56675091 IC50 = 2.2 nM T98691 CA2Z0U 56676986 IC50 = 58.5 nM T98691 CX0FH5 56678398 IC50 = 30 nM T98691 C3WEQ5 56678399 IC50 = 1.9 nM T98691 CD67LW 56678400 IC50 = 2.2 nM T98691 C24QMN 56680316 IC50 = 4400 nM T98691 CX8M7Z 56683636 IC50 = 4.8 nM T98691 CK5X0U 57619789 IC50 > 10000 nM T98691 CH3M0B 59543520 IC50 > 25000 nM T98691 CCR9Q8 59543629 IC50 = 8300 nM T98691 C3ESJ1 59543757 IC50 = 6800 nM T98691 CZV45P 59619390 IC50 > 25000 nM T98691 C75LIT 59907274 Ki = 27 nM T98691 CLX2Y4 60148518 Ki = 37000 nM T98691 C0DA6M 60166364 Ki > 40000 nM T98691 C4G1SF 60166365 Ki > 40000 nM T98691 COM7U3 60166366 Ki > 4000 nM T98691 COQ82A 60166367 Ki > 4000 nM T98691 C2Y7EK 60166492 Ki > 4000 nM T98691 C4PHR1 60166493 Ki > 4000 nM T98691 CG4DZ7 60166494 Ki > 4000 nM T98691 C5E2PB 60166495 Ki > 4000 nM T98691 CXD39V 60166496 Ki > 4000 nM T98691 CM8XO5 60166497 Ki > 4000 nM T98691 C7XLR3 60169906 Ki = 200 nM T98691 CA95CZ 60195809 IC50 > 40000 nM T98691 CY3VC4 60195810 IC50 > 100000 nM T98691 CMA8T3 60195811 IC50 > 100000 nM T98691 CVRJ91 60195812 IC50 = 3110 nM T98691 CE6AH0 60195813 IC50 > 40000 nM T98691 C8ILH6 60195902 IC50 > 10000 nM T98691 CX4N2V 60195903 IC50 > 40000 nM T98691 C4PQ6E 60195904 IC50 > 100000 nM T98691 CNUI89 60195905 IC50 > 40000 nM T98691 C23JUZ 60195906 IC50 > 100000 nM T98691 CBY72G 66572720 Ki = 1500 nM T98691 C34GCU 66572722 IC50 = 16000 nM T98691 CHWA75 66572723 IC50 = 8600 nM T98691 C78CAD 66572724 IC50 = 9000 nM T98691 CAF7U2 66572726 Ki = 900 nM T98691 C3V1BY 66572849 IC50 = 1100 nM T98691 C1Q5WX 66572850 IC50 = 13000 nM T98691 CLJ58E 66572851 Ki = 200 nM T98691 C3VLY0 66572852 IC50 = 19300 nM T98691 C4TXD6 66572853 IC50 = 1500 nM T98691 CJOF37 67298501 Ki = 794.33 nM T98691 C6P9GX 68485393 IC50 = 20000 nM T98691 C4JPF2 69924862 IC50 = 1000 nM T98691 CBR31D 69925026 IC50 = 1300 nM T98691 CVJ5F3 69925527 IC50 = 500 nM T98691 CSF35K 70274227 IC50 > 10000 nM T98691 CI0XF8 70274815 IC50 > 100000 nM T98691 CXT5G7 70275845 IC50 > 10000 nM T98691 C5P3BO 70275923 IC50 > 10000 nM T98691 CCG16F 70276365 IC50 > 100000 nM T98691 C0T3LC 70276605 IC50 > 10000 nM T98691 CE1J0O 70276811 IC50 > 100000 nM T98691 C06WFN 70276830 IC50 > 100000 nM T98691 CDQ85E 70276990 IC50 = 10000 nM T98691 CGET13 70278898 IC50 > 10000 nM T98691 C2GT5H 70280758 IC50 > 100000 nM T98691 CI53XU 70281040 IC50 > 10000 nM T98691 CA6DM2 70281073 IC50 > 100000 nM T98691 CS8VR4 70676096 Ki = 1330 nM T98691 CJQX06 70681840 IC50 = 3600 nM T98691 CW8L0K 70682252 IC50 = 1500 nM T98691 C1UIK4 70682253 IC50 = 284 nM T98691 CSW1R7 70682254 IC50 = 256 nM T98691 CY2WE3 70682255 IC50 > 10000 nM T98691 CVHX94 70682256 IC50 > 10000 nM T98691 CNF23Q 70682257 IC50 = 112 nM T98691 CZ84UX 70682584 IC50 > 100000 nM T98691 CR45PO 70683941 IC50 = 26000 nM T98691 CZI74Q 70683995 IC50 = 26000 nM T98691 CADN96 70683996 IC50 > 50000 nM T98691 C8S1DB 70684341 IC50 > 10000 nM T98691 CH7L2N 70684342 IC50 > 10000 nM T98691 CM5C8Q 70686123 Ki = 1900 nM T98691 CN4QX8 70686124 IC50 = 11000 nM T98691 CM2V0E 70686501 IC50 = 2720 nM T98691 CSPH68 70686502 IC50 > 10000 nM T98691 CL9RE3 70686820 IC50 > 100000 nM T98691 C65EDY 70686822 IC50 > 100000 nM T98691 CBV9F6 70688255 IC50 = 7200 nM T98691 C47WPT 70688256 IC50 = 3200 nM T98691 CMW4T8 70688257 IC50 = 5700 nM T98691 CWE9C8 70688597 IC50 = 46 nM T98691 CV20NB 70688598 IC50 > 10000 nM T98691 CJ4FO1 70688599 IC50 = 1117 nM T98691 CIR23C 70688600 IC50 > 10000 nM T98691 C5NMF8 70688601 IC50 > 10000 nM T98691 C5IYR0 70688897 IC50 > 100000 nM T98691 CA1Q0F 70690660 IC50 = 68 nM T98691 CZY5R0 70690661 IC50 > 10000 nM T98691 C2Z8JP 70690662 IC50 > 10000 nM T98691 C73CZT 70690663 IC50 = 6521 nM T98691 C2H1NL 70690664 IC50 = 260 nM T98691 CLE18H 70692439 IC50 = 2500 nM T98691 CAB1L6 70692440 Ki = 1900 nM T98691 C5D8SA 70692441 IC50 > 50000 nM T98691 CE8Q4U 70692809 IC50 = 434 nM T98691 CND37B 70692810 IC50 > 10000 nM T98691 CZOF81 70693115 IC50 > 100000 nM T98691 CMFW03 70693116 IC50 > 100000 nM T98691 C5RSJ0 70693117 IC50 > 100000 nM T98691 C36JBX 70694841 IC50 > 10000 nM T98691 C86ETZ 70694842 IC50 > 10000 nM T98691 CAU9C4 70694843 IC50 = 3650 nM T98691 C4A7HL 70694844 IC50 = 3960 nM T98691 C01IDC 70695171 IC50 > 100000 nM T98691 CGV1W9 70696541 IC50 > 50000 nM T98691 CXY0A7 70696542 IC50 = 18200 nM T98691 C8HEM6 70696892 IC50 = 214 nM T98691 CK5RP0 70696893 IC50 > 10000 nM T98691 C34WHG 70697225 IC50 > 100000 nM T98691 C0H1BV 70788951 IC50 > 250000 nM T98691 CS60PU 71450699 IC50 = 200 nM T98691 CS58YC 71450700 IC50 = 400 nM T98691 C08LGJ 71451733 IC50 > 10000 nM T98691 CI7Z8B 71451734 IC50 > 10000 nM T98691 C2UN6D 71452029 IC50 > 100000 nM T98691 CG8T7Z 71452030 IC50 > 100000 nM T98691 C7RJG8 71453558 IC50 > 10000 nM T98691 C2OGP1 71453559 IC50 > 10000 nM T98691 CDR10X 71453560 IC50 > 10000 nM T98691 CZ6M8U 71454284 IC50 = 600 nM T98691 CP7H6S 71454285 IC50 > 20000 nM T98691 CFUS41 71455276 IC50 > 10000 nM T98691 CUQL74 71455277 IC50 > 10000 nM T98691 C0KUW5 71455278 IC50 > 10000 nM T98691 C7Z0HF 71455279 IC50 > 10000 nM T98691 C78BKL 71455561 IC50 > 100000 nM T98691 C9YJG7 71457065 IC50 > 10000 nM T98691 C3IH8Z 71457841 IC50 = 18000 nM T98691 CCH47M 71458921 IC50 > 10000 nM T98691 CP7MZ5 71458922 IC50 > 10000 nM T98691 CCA46N 71458923 IC50 > 10000 nM T98691 CQT1C2 71458924 IC50 > 10000 nM T98691 CZT23D 71459213 IC50 = 10800 nM T98691 CF69OZ 71459754 IC50 = 50 nM T98691 CDW0I7 71460731 IC50 > 10000 nM T98691 CC87WL 71460732 IC50 > 10000 nM T98691 CL6Y4C 71460733 IC50 > 10000 nM T98691 C7GX8H 71463202 IC50 = 130 nM T98691 CZM3L7 71520324 Ki = 124000 nM T98691 C5YQ6V 71602930 IC50 > 10000 nM T98691 CY7EL9 71602931 IC50 > 10000 nM T98691 CC61PX 71602932 IC50 > 10000 nM T98691 CH5QG3 71602933 IC50 > 10000 nM T98691 COU6R5 71602979 IC50 > 10000 nM T98691 CR6JV1 71602981 IC50 > 10000 nM T98691 CP87FL 71602983 IC50 = 1740 nM T98691 C34RLW 71602984 IC50 > 10000 nM T98691 CL6B0E 71602986 IC50 > 10000 nM T98691 CQ1ZN0 71603042 IC50 = 658 nM T98691 C6SWY5 71603043 IC50 >= 10000 nM T98691 CD0Z4V 71603045 IC50 > 10000 nM T98691 C1YCF7 71603046 IC50 > 10000 nM T98691 C2VH5F 71603047 IC50 > 10000 nM T98691 CQ76CG 71603106 IC50 > 10000 nM T98691 CF9J1B 71603109 IC50 > 10000 nM T98691 CMSE93 71603111 IC50 > 10000 nM T98691 CIU41Z 71603112 IC50 > 10000 nM T98691 C9GMP4 71603168 IC50 = 228 nM T98691 CSI94H 71612693 Ki = 1700 nM T98691 CH65CP 71612694 Ki = 2600 nM T98691 CER82H 71612695 Ki = 120 nM T98691 C3WV1B 71612696 Ki = 1000 nM T98691 CJ71KZ 71612697 Ki = 20000 nM T98691 COZ0E4 71612901 Ki = 9000 nM T98691 CQ3XD4 71612902 Ki = 1000 nM T98691 C4U0TK 71612903 Ki = 2900 nM T98691 CA82UN 71612904 Ki = 2300 nM T98691 CY02ME 71612905 Ki = 2400 nM T98691 C4TG6P 71612906 Ki = 2600 nM T98691 C3PY2W 71613098 Ki = 2700 nM T98691 C7KF1W 71613099 Ki = 6800 nM T98691 CAG6F9 71613100 Ki = 5500 nM T98691 CI0Q7G 71613101 Ki = 5000 nM T98691 CTH19S 71613102 Ki = 4600 nM T98691 CV60XA 71613103 Ki = 6100 nM T98691 C90OHP 71613322 Ki = 7800 nM T98691 CRP54C 71613323 Ki = 3200 nM T98691 C85WJH 71613324 Ki = 2500 nM T98691 C6HK4W 71615678 Ki = 2400 nM T98691 C7CN4G 71615679 Ki = 1800 nM T98691 C8JN2W 71615680 Ki = 1700 nM T98691 CN32FZ 71615681 Ki = 2500 nM T98691 C4XUV9 71615682 Ki = 23000 nM T98691 CNZ0K4 71624621 IC50 = 67510 nM T98691 C9QY7K 71624622 IC50 = 45270 nM T98691 C0S6HT 71624732 IC50 > 100000 nM T98691 C3CRY6 71624733 IC50 = 73220 nM T98691 C37EVT 71624734 IC50 = 39310 nM T98691 C9P1QH 71624735 IC50 = 91170 nM T98691 CNCX24 71624736 IC50 = 4720 nM T98691 CI5T0R 71656572 Ki = 2.4 nM T98691 CAN6X5 71656574 Ki = 10 nM T98691 C4I0VB 71656669 Ki = 3 nM T98691 CH2J8G 71663299 Ki = 13 nM T98691 C63ROI 71717313 Ki = 155000 nM T98691 C0JYT2 71717876 IC50 = 160 nM T98691 COZB76 71720328 IC50 = 300 nM T98691 C05PXN 71720329 IC50 = 130 nM T98691 C0O5NF 71726670 IC50 = 9.85 nM T98691 CW16QR 71738813 IC50 = 8.12 nM T98691 CS31TK 71738883 IC50 = 14.4 nM T98691 CIO7K3 73345851 Ki = 26000 nM T98691 CY1IU2 73345852 Ki = 390 nM T98691 CDQP51 73347119 Ki = 15000 nM T98691 CJQE58 73348851 Ki = 4200 nM T98691 C5XOV2 73348852 Ki = 27000 nM T98691 C31JUR 73348857 Ki = 740 nM T98691 C95BEA 73348858 Ki = 890 nM T98691 CM3PH8 73350210 Ki = 146000 nM T98691 CZN1M9 73350437 Ki = 3500 nM T98691 CMD57T 73350441 Ki = 7000 nM T98691 CBO54W 73351952 Ki = 28000 nM T98691 COC70E 73351953 Ki = 14000 nM T98691 CAYM96 73351955 Ki = 450 nM T98691 CXR1B9 73353408 Ki = 1400 nM T98691 CNQA65 73354924 Ki = 2600 nM T98691 C37HIQ 73354926 Ki = 3100 nM T98691 CJ6CQ1 73356205 Ki = 400 nM T98691 CL37SD 73356439 IC50 > 10000 nM T98691 CYSR74 73356489 Ki = 4200 nM T98691 CW9NU4 73895627 Ki = 27 nM T98691 CIE28G 73895715 IC50 = 1200 nM T98691 CO68XU 73895952 IC50 = 190 nM T98691 CK3U8P 77907483 IC50 = 2200 nM T98691 CR05TU 89809888 IC50 = 654 nM T98691 CHJB16 89886996 IC50 = 56 nM T98691 CIXT20 89888879 IC50 = 23.8 nM T98691 C62SML 90655967 IC50 > 10000 nM T98691 CJ7LT3 90655968 IC50 > 10000 nM T98691 CB61WC 90655969 IC50 > 10000 nM T98691 CIS56R 90663177 Ki = 720 nM T98691 CU71EO 90663180 Ki = 1000 nM T98691 CX37IK 90663181 Ki = 18 nM T98691 CM4GY1 90663406 Ki = 210 nM T98691 CSD0G2 90663407 Ki = 21 nM T98691 C5F0JO 90663408 Ki = 200 nM T98691 CTNU67 90663409 Ki = 490 nM T98691 CX9NC2 90663410 Ki = 270 nM T98691 CV97ET 90663411 Ki = 3900 nM T98691 CJ2V9B 90663412 Ki = 45 nM T98691 CEZ3N7 90663413 Ki = 240 nM T98691 C7SBR9 90663414 Ki = 270 nM T98691 C9KYG2 90663415 Ki = 160 nM T98691 C7PZ8K 90663416 Ki = 16 nM T98691 C89DWE 90663417 Ki = 67 nM T98691 CX9I6Z 90663418 Ki = 19 nM T98691 C9MQ4F 90663419 Ki = 6600 nM T98691 C0FO3U 90663420 Ki = 210 nM T98691 CF29CP 90663422 Ki = 38000 nM T98691 CJH31Z 90665726 Ki = 25100 nM T98691 CX7WG9 90665730 Ki = 29800 nM T98691 CFKB46 90665732 Ki = 13100 nM T98691 CB14DH 90665735 Ki = 820 nM T98691 C0XZH3 90665919 IC50 = 5870 nM T98691 C0HIA4 90665921 IC50 = 4390 nM T98691 C5AIN7 91667613 IC50 > 10000 nM T98691 CH68BZ 91885514 Ki = 720 nM T98691 CRVO29 91885636 Ki = 11000 nM T98691 CGFK60 101201806 IC50 = 25500 nM T98691 CK0AF8 101889645 IC50 > 100000 nM T98691 C7I4XF 101889646 IC50 > 100000 nM T98691 C8E4WS 102323332 IC50 = 29500 nM T98691 CVJF59 118716317 Ki = 573 nM T98691 CA79YF 118716318 Ki = 228 nM T98691 C3Q5BM 118716319 Ki = 185 nM T98691 CI6H0V 118716320 Ki = 1690 nM T98691 CL4ES1 118716560 IC50 > 100000 nM T98691 C5ALU2 118719334 IC50 = 3300 nM T98691 CTE34I 118720232 IC50 > 100000 nM T98691 CSD62B 118720233 IC50 = 100000 nM T98691 C9WF7Q 118720234 IC50 = 5600 nM T98691 C76HIO 118720235 IC50 > 11000 nM T98691 CAT1R6 118720236 IC50 > 100000 nM T98691 CGAF42 118720237 IC50 > 100000 nM T98691 CJ28KZ 118720238 IC50 > 100000 nM T98691 CPH2V9 118720239 IC50 > 100000 nM T98691 CMBG29 118724585 IC50 = 1000 nM T98691 C35TQG 122186479 Ki = 10000 nM T98691 CF0CG5 122186480 Ki = 1200 nM T98691 CV46XN 122194107 IC50 = 1522 nM T98691 CYO0X5 122194108 IC50 > 10000 nM T98691 CW6K0Z 122194109 IC50 = 5117 nM T98691 CO02XD 122194111 IC50 = 10000 nM T98691 CT51QX 122194112 IC50 = 71.6 nM T98691 CYLN40 122194113 IC50 = 10347 nM T98691 CRS8C6 126610725 IC50 > 10000 nM T98691 CN2IE8 126610758 IC50 >= 10000 nM T98691 C2E4BP 126610767 IC50 >= 10000 nM T98691 C2HJS3 126610779 IC50 > 10000 nM T98691 C2ZL3O 126610781 IC50 > 10000 nM T98691 CJV56I 126610782 Ki = 8.4 nM T98691 CMT2B9 127049869 Ki = 1.27 nM T98691 C43APM 127050163 Ki = 2160 nM T98691 C8VKA5 127050164 Ki = 1920 nM T98691 CZ54XC 127050165 Ki = 431 nM T98691 CI2C3V 127050166 Ki = 6300 nM T98691 CY3JP6 127050263 EC50 = 6000 nM T98691 C7V8XZ 127051317 Ki = 6980 nM T98691 CSK16Q 127051318 Ki = 11700 nM T98691 C7YI4M 127051342 Ki = 4300 nM T98691 C6NFU9 127051343 Ki = 609 nM T98691 C6SD7P 127051344 Ki = 707 nM T98691 CY5CV6 127051345 Ki = 1050 nM T98691 C7HX5O 127054405 IC50 = 320 nM T98691 CEC17N 129164665 Ki = 143 nM T98691 CF9WE3 129164666 Ki = 1522 nM T98691 CY4B7Z 129164668 Ki = 15 nM T98691 CF03SH 129164670 Ki = 181 nM T98691 CEG65P 129164672 Ki = 11 nM T98691 CBSX69 129164675 Ki = 1116 nM T98691 CJO2P0 129164678 Ki = 25 nM T98691 CL9RX5 129164679 Ki = 14 nM T98691 C10YQZ 129164681 Ki = 181 nM T98691 COT2J5 129164699 Ki = 4 nM T98691 CSLH25 129164700 Ki = 1473 nM T98691 CAT90Y 129164701 Ki = 353 nM T98691 CSG89A 129164702 Ki = 82 nM T98691 C89OZL 129164715 Ki = 82 nM T98691 CJ7T4Z 129164725 Ki = 81.7 nM T98691 C3Q5VE 129164742 Ki = 112 nM T98691 CUB58Q 129164743 Ki = 266 nM T98691 CBC15M 129164750 Ki = 76 nM T98691 CS85KM 129164773 Ki = 314 nM T98691 CPG69E 129178768 Ki = 93 nM T98691 CK6I7U 129178772 Ki = 64 nM T98691 C94NGL 129178773 Ki = 7 nM T98691 C41ZCQ 129178794 Ki = 78 nM T98691 CD1I3P 129178829 Ki = 1076 nM T98691 C81SHO 129178830 Ki = 8 nM T98691 CV2LA1 129178843 Ki = 467 nM T98691 C8SD2H 134132002 Ki = 280 nM T98691 C2CT4O 134134083 IC50 = 45 nM T98691 C0U6GR 134134734 Ki = 110 nM T98691 CD5NI4 134134799 Ki = 11 nM T98691 CE53MB 134135884 Ki = 2020 nM T98691 CD0UE9 134136855 IC50 = 17 nM T98691 CW3B7G 134137121 Ki = 49 nM T98691 CF8VA4 134138144 IC50 = 17 nM T98691 C4CT5Z 134139989 Ki = 46 nM T98691 CQ8U5W 134141808 IC50 = 113 nM T98691 C3PEW2 134141970 IC50 = 136 nM T98691 CV36BU 134142724 IC50 = 226 nM T98691 C4BXO1 134144535 IC50 = 23 nM T98691 C4HN8V 134148867 Ki = 30 nM T98691 CH98KJ 134154138 Ki = 19.6 nM T98691 C4TS3J 134154893 IC50 = 17 nM T98691 C2UMT4 134157443 Ki = 200 nM T98691 CEU25N 135137860 Ki = 59000 nM T98691 C5DI9L 135285655 Ki = 253 nM T98691 CNEY95 135285657 Ki = 131 nM T98691 CUVL51 135872798 IC50 = 164 nM T98691 CA8Y4C 136002680 IC50 > 10000 nM T98691 CTQY96 136117851 IC50 = 10 nM T98691 CH08TX 136218747 IC50 > 10000 nM T98691 C2DF5Q 136218748 IC50 > 10000 nM T98691 CL46RX 136218749 IC50 = 449 nM T98691 CGR2E9 136218750 IC50 = 338 nM T98691 CRUC19 137028456 IC50 = 340.5 nM T98691 CS9BV2 137631536 Ki = 1.2 nM T98691 CF94BI 137631849 Ki = 443 nM T98691 CXFL83 137632292 Ki = 217 nM T98691 C13NEP 137633621 Ki = 1430 nM T98691 C23MHJ 137633661 Ki > 5100 nM T98691 CIQ6J5 137633888 Ki = 824 nM T98691 C98CSB 137634116 Ki = 4.6 nM T98691 CBH9O3 137634490 Ki = 2790 nM T98691 CNJ09U 137634671 Ki = 2.5 nM T98691 CI52RD 137635205 Ki = 676 nM T98691 C7Y6UT 137635495 Ki = 7.3 nM T98691 CT5X3N 137635933 Ki = 12 nM T98691 CDF39A 137636254 Ki = 123 nM T98691 CLC04W 137636315 Ki = 1105.7 nM T98691 CG6MH5 137636590 Ki = 30 nM T98691 CT39DN 137637025 Ki = 240 nM T98691 C39AXE 137637300 Ki = 2.2 nM T98691 C7RZ4Q 137638604 Ki = 77 nM T98691 C5MF9X 137638638 Ki = 250 nM T98691 CVJU21 137638762 Ki > 5100 nM T98691 C4W7BD 137638856 Ki = 3860 nM T98691 C25QTS 137639741 Ki = 110 nM T98691 CIZ32F 137639823 IC50 > 10000 nM T98691 CW7IU5 137639903 Ki = 1750 nM T98691 CLX0W9 137640185 Ki = 55.7 nM T98691 CF2QB8 137641334 Ki > 20000 nM T98691 CPV52Z 137641366 Ki > 5100 nM T98691 CO28QB 137642402 Ki = 5.8 nM T98691 CQY6I2 137642965 Ki = 3.7 nM T98691 CVXI65 137643204 Ki = 1364.2 nM T98691 C62IJM 137643751 Ki = 997 nM T98691 CQ98DG 137644516 Ki > 5100 nM T98691 CNS6X7 137644585 Ki = 952 nM T98691 CZC96S 137645782 Ki = 6393.3 nM T98691 CKUJ94 137646266 Ki = 91 nM T98691 C9P6IF 137646532 Ki > 5100 nM T98691 C0TUX3 137646586 Ki = 167 nM T98691 CB7Q5U 137646785 Ki = 7.4 nM T98691 C1AXD7 137647008 Ki = 0.61 nM T98691 CU7BJ0 137647125 Ki = 1.2 nM T98691 CM3OP2 137647368 Ki = 5100 nM T98691 C9F0MH 137647486 Ki = 3020 nM T98691 CZK74L 137647856 Ki = 45 nM T98691 C8FS0C 137649214 Ki = 411 nM T98691 C86ZJA 137649575 Ki = 279 nM T98691 CV54KX 137651518 Ki = 3500 nM T98691 CZBU13 137651934 Ki = 0.4 nM T98691 C4SO3J 137652485 Ki = 1800 nM T98691 CGY3U7 137653100 Ki = 77 nM T98691 CS8U7B 137653242 Ki = 25 nM T98691 CD9P4B 137653316 Ki = 1010 nM T98691 CN79HC 137653449 Ki = 15.5 nM T98691 C4WBO2 137654260 Ki = 505 nM T98691 CG75LU 137654285 Ki = 273.5 nM T98691 C48MPO 137655059 Ki = 1020 nM T98691 C5VI1O 137655103 Ki = 40.3 nM T98691 CR7I0L 137655469 Ki > 5100 nM T98691 C5QVE7 137655537 Ki = 3.5 nM T98691 CB1X4P 137656245 Ki = 304 nM T98691 C6RJO9 137656888 Ki = 25 nM T98691 C4F5SL 137658767 Ki = 671 nM T98691 CZA12J 137659286 Ki = 330 nM T98691 CPA9N7 137659410 Ki > 5100 nM T98691 CL2BY4 137659508 Ki = 5.6 nM T98691 C17LXI 137660025 Ki = 2.3 nM T98691 CT9PH8 137660357 IC50 = 8550 nM T98691 C2FGL6 137660813 Ki = 40 nM T98691 CVP27L 137661274 Ki = 358 nM T98691 C6MI1F 137661465 Ki = 41 nM T98691 CU05SB 137662237 Ki = 515 nM T98691 CEW35U 137662313 Ki = 27 nM T98691 C8A2PN 145960387 IC50 = 92 nM T98691 CFD97H 145960437 IC50 = 2500 nM T98691 C2ER0T 145961056 IC50 = 140 nM T98691 CNJ1G2 145961256 IC50 = 86 nM T98691 C2NFQ1 145961390 IC50 = 110 nM T98691 CAGM09 145961698 IC50 = 1200 nM T98691 C5SLU2 145961778 IC50 = 3500 nM T98691 CIUS59 145962186 IC50 = 280 nM T98691 C3LZB4 145962243 IC50 = 15 nM T98691 CXJ82U 145962422 IC50 = 84 nM T98691 CWYS01 145962673 IC50 = 130 nM T98691 CF8E2T 145962685 IC50 = 4100 nM T98691 CLF40P 145962976 IC50 = 42 nM T98691 CS85OZ 145963002 IC50 = 240 nM T98691 CLP70J 145963229 IC50 = 816000 nM T98691 CY83PE 145963309 IC50 = 140 nM T98691 CSMC76 145963498 IC50 = 590 nM T98691 CJ38RF 145963551 IC50 = 77 nM T98691 C75PCG 145963584 IC50 = 93 nM T98691 CMN91X 145963645 IC50 = 48 nM T98691 CO6UD2 145963721 IC50 = 280 nM T98691 CFQ25D 145967499 IC50 = 755 nM T98691 CIVB10 145967715 IC50 = 4 nM T98691 CLI6T0 145967952 IC50 = 2630 nM T98691 CC4AG7 145968405 IC50 > 5000 nM T98691 CDS31M 145968622 IC50 = 492 nM T98691 CA40YU 145969275 IC50 = 635 nM T98691 CB0Y7Z 145969438 IC50 > 5000 nM T98691 C2WCK0 145969450 IC50 = 300 nM T98691 CL7KO9 145969878 IC50 > 5000 nM T98691 C3NAS7 145970030 IC50 > 5000 nM T98691 C8X6JG 145970039 Ki = 195000 nM T98691 C51ZEH 145970706 Ki = 155000 nM T98691 CS08XI 145970918 IC50 > 5000 nM T98691 C9XKW2 145970931 IC50 = 494 nM T98691 CQ3TG0 145979639 Ki = 22000 nM T98691 CXW3F1 145982578 IC50 = 400 nM T98691 CY7XE4 145982644 IC50 = 4600 nM T98691 C56AXR 145982654 IC50 = 62000 nM T98691 CNC48W 145982661 IC50 = 210 nM T98691 CMS4E9 145982820 IC50 = 260 nM T98691 C7S2TX 145983004 IC50 = 500 nM T98691 CU5Z9F 145983387 IC50 = 2450 nM T98691 CWA21O 145983581 IC50 = 14300 nM T98691 C1OEA0 145983615 IC50 = 500 nM T98691 C6JSW3 145983652 IC50 = 50 nM T98691 C7V2ZF 145983823 IC50 = 1300 nM T98691 CV8HP6 145984203 Ki = 5 nM T98691 C3JIQ4 145984217 IC50 = 18000 nM T98691 CT8QM9 145984597 IC50 = 9500 nM T98691 C3LH7B 145984676 IC50 = 10 nM T98691 CUT36M 145984739 IC50 = 13100 nM T98691 CJM6L4 145984752 IC50 = 400 nM T98691 C0BC2Z 145984777 IC50 = 5300 nM T98691 CJK42D 145985003 IC50 = 180 nM T98691 CGC54P 145985016 IC50 = 1400 nM T98691 C8AM0K 145985030 IC50 = 1490 nM T98691 CURI53 145985037 IC50 = 10 nM T98691 C2LB8K 145985094 IC50 = 200 nM T98691 CNT63X 145985191 IC50 = 30 nM T98691 CHCP90 145985556 IC50 > 2000 nM T98691 CX6JT1 145985564 IC50 = 600 nM T98691 CJE7L9 145985615 IC50 = 37000 nM T98691 CL2B3Y 145985677 IC50 = 1300 nM T98691 C9C5YA 145985785 IC50 = 47000 nM T98691 CBK3G5 145985888 IC50 = 90 nM T98691 CQ2RS8 145986120 IC50 = 1600 nM T98691 CM53FT 145986712 Ki = 5 nM T98691 C6OKB9 145987263 IC50 > 5000 nM T98691 CRD65W 145987430 Ki = 30000 nM T98691 COZ6P5 145987960 IC50 = 4275 nM T98691 C7ZCW3 145988622 IC50 = 334 nM T98691 CN6U8D 145988823 Ki = 5000 nM T98691 C9OAK6 145989037 IC50 = 99 nM T98691 C87GKT 145989707 IC50 = 1591 nM T98691 C8NW1T 145990306 Ki = 12000 nM T98691 C5MWT1 145990477 Ki = 2000 nM T98691 CH7WO9 145994261 Ki = 7300 nM T98691 CUAY08 148018738 IC50 = 3000 nM T98691 CQK39B 149491764 IC50 > 10000 nM T98691 C1ZX5D 149494192 IC50 = 3000 nM T98691 CJ2DW5 155510635 Ki = 1000 nM T98691 CKT12D 155510715 Ki = 1900 nM T98691 CK8F2Z 155512199 Ki = 14.8 nM T98691 COR3E2 155513054 Ki = 10.2 nM T98691 CFN98D 155513234 Ki = 453 nM T98691 CF01VN 155514418 Ki = 630.96 nM T98691 CK6AQ2 155514722 Ki = 398.11 nM T98691 C27SKJ 155515029 IC50 = 0.094 nM T98691 C8HP4U 155515082 Ki > 10000 nM T98691 C6L2RD 155515575 Ki = 230 nM T98691 CJ6Z4N 155515766 Ki = 19.95 nM T98691 CWDS96 155516109 Ki = 47 nM T98691 C5U6FM 155517896 IC50 = 1.35 nM T98691 CYL03V 155518363 Ki = 251.19 nM T98691 CKJ9V2 155519071 IC50 = 0.632 nM T98691 CT94JP 155519833 Ki = 125.89 nM T98691 CE76XY 155520224 Ki = 100 nM T98691 CBK28U 155521458 Ki = 158.49 nM T98691 C0EWD4 155522491 Ki = 5.012 nM T98691 CI9YP3 155522753 Ki = 47 nM T98691 CO2Y0C 155523098 Ki = 700 nM T98691 CZ3KD7 155523939 Ki = 90.3 nM T98691 CBN12I 155524050 Ki = 406 nM T98691 CZI5G3 155524425 Ki = 78.2 nM T98691 C6M1FK 155524435 Ki = 1584.89 nM T98691 CC9X2D 155525224 Ki = 251.19 nM T98691 CD7WG5 155525553 IC50 = 6.64 nM T98691 CNLO46 155526163 Ki = 158.3 nM T98691 CL57AH 155526723 Ki = 108.2 nM T98691 CZ0A5X 155527224 Ki = 158.49 nM T98691 C16ZBY 155529633 Ki = 501.19 nM T98691 C87DAI 155530185 Ki = 39.81 nM T98691 CVN4I3 155530380 Ki = 174.8 nM T98691 C0WZD4 155533248 IC50 = 376 nM T98691 C92YHN 155535180 IC50 = 1.31 nM T98691 CZ59GS 155536157 Ki = 25.12 nM T98691 CB4MT7 155537119 IC50 = 1.68 nM T98691 CYA0Q2 155537428 Ki = 1.5 nM T98691 CNMR90 155537964 IC50 = 3.54 nM T98691 CXHT61 155539577 IC50 = 77 nM T98691 CTV4B7 155539870 IC50 = 1.73 nM T98691 CFRP81 155539888 Ki = 1000 nM T98691 C26AMH 155539986 Ki = 5.3 nM T98691 C95CPE 155540752 Ki = 146000 nM T98691 CO3ZF7 155541809 Ki = 880 nM T98691 C47OMS 155542219 Ki = 100 nM T98691 C43ZKT 155544277 IC50 = 3.53 nM T98691 CB94ZI 155544429 IC50 = 3.13 nM T98691 CIZ8A6 155544625 IC50 = 0.79 nM T98691 CQW2L9 155545346 Ki = 1584.89 nM T98691 CY2TK7 155547967 Ki = 1258.93 nM T98691 CXYT09 155551122 Ki = 195 nM T98691 CT7P2Z 155551886 Ki = 251.19 nM T98691 C3TS9N 155552318 Ki = 158.49 nM T98691 CCF86H 155553085 Ki = 4300 nM T98691 C8Z7GU 155553621 Ki = 630.96 nM T98691 CF0X8Z 155554135 Ki = 199.53 nM T98691 C2P9GA 155554760 IC50 = 47 nM T98691 C6O9FK 155556968 Ki = 1100 nM T98691 C2AIC6 155559777 IC50 = 4.15 nM T98691 CPCR48 155561105 Ki = 35 nM T98691 CRO9V2 155561992 IC50 = 1 nM T98691 CA6XR1 155562235 Ki = 251.19 nM T98691 C1N3AJ 155565629 Ki = 63.1 nM T98691 C3Z7UC 155566273 Ki = 0.6 nM T98691 CW30IO 155567009 Ki = 630.96 nM T98691 CFTW36 155567371 Ki = 76 nM T98691 CLOJ91 155567513 Ki = 4.1 nM T98691 CHD79T 44408017 IC50 = 14000 nM T98691 CO0N3S 44408050 IC50 = 3400 nM T98691 C58OLD 44517711 IC50 = 1.995 nM T98691 CT3S1I 44517712 IC50 = 1.259 nM T98691 CFT38D 45267632 IC50 = 15.85 nM T98691 COU83P 45267640 IC50 = 199.53 nM T98691 C1U4IF 45267645 IC50 = 125.89 nM T98691 CDG5S8 45268499 IC50 = 501.19 nM T98691 CV8PZ3 45268510 IC50 > 7943.28 nM T98691 C89ADF 45269361 IC50 = 794.33 nM T98691 C58PZI 45269375 IC50 = 501.19 nM T98691 C5O9EF 45270206 IC50 = 5.012 nM T98691 C07ADH 45270207 IC50 = 3.981 nM T98691 CVGE81 45270212 IC50 = 6.31 nM T98691 C78EXG 45271021 IC50 = 1995.26 nM T98691 C5MBC4 45271038 IC50 = 5.012 nM T98691 C65QLD 45271887 IC50 = 3981.07 nM T98691 CIL8O6 45271888 IC50 = 1584.89 nM T98691 CLFD35 45272742 IC50 = 3162.28 nM T98691 C3WF8S 45272748 IC50 = 3162.28 nM T98691 CQO98K 45272752 IC50 = 1258.93 nM T98691 C9A0IH 45272753 IC50 = 15.85 nM T98691 CSYU09 45273681 IC50 = 1584.89 nM T98691 C0HRW4 70690665 IC50 > 10000 nM T98691 CU60DG 70696894 IC50 > 10000 nM T98691 D00FGA 73737 IC50 = 1584.89 nM T98691 D00VAN 46232847 IC50 = 224 nM T98691 D01CSE 52942034 IC50 = 232.4 nM T98691 D03JYN 15722900 IC50 = 1020 nM T98691 D04BGT 46881451 IC50 > 10000 nM T98691 D04DFX 136002679 IC50 = 126.1 nM T98691 D05WZF 10129151 IC50 > 5000 nM T98691 D06WQP 60148519 Ki = 15 nM T98691 D08KCA 72429 IC50 = 2.5 nM T98691 D08TMM 9851116 IC50 = 0.2 nM T98691 D08TWJ 10095492 Ki = 970 nM T98691 D09FGQ 123985 IC50 = 13 nM T98691 D09NBP 52940642 IC50 = 1000 nM T98691 D0B2FE 46882093 IC50 > 10000 nM T98691 D0B2JC 46232967 IC50 = 2160 nM T98691 D0B4JS 44449925 IC50 = 910 nM T98691 D0D0JU 14849212 Ki = 10400 nM T98691 D0D0LD 9913088 IC50 = 1221 nM T98691 D0G2QG 44343301 IC50 = 740 nM T98691 D0G8OD 11702208 Ki = 2790 nM T98691 D0J7OM 24777047 IC50 = 4380 nM T98691 D0LL1F 52945875 IC50 = 5410 nM T98691 D0M3AP 46232386 IC50 = 4870 nM T98691 D0MD6D 24778186 IC50 = 12220 nM T98691 D0R2BO 194777 IC50 > 1000 nM T98691 D0S4EI 10244468 Ki = 31700 nM T98691 D0T0IR 49865939 Ki = 3400 nM T98691 D0T7QF 10420833 IC50 = 8900 nM T98691 D0V7LZ 74761 Ki = 11300 nM T98691 D0VE0F 10062714 IC50 = 2000 nM T98691 D0X9YD 65036 Ki = 9300 nM T98691 D0Z0PR 9912381 IC50 = 340 nM T87831 D0G7UX 5284373 IC50 > 10000 nM T87831 CH35QD 125628 IC50 = 2000 nM T87831 C1EC2Q 457933 EC50 = 500 nM T87831 CNHO18 3089940 IC50 = 1258.93 nM T87831 CVK6F2 3825824 IC50 = 2511.89 nM T87831 C5CE6R 3939767 IC50 = 316.23 nM T87831 CRU1E6 4652862 IC50 = 2511.89 nM T87831 C3BMC2 4654636 IC50 = 794.33 nM T87831 CYGD06 4881668 IC50 = 3981.07 nM T87831 CZY10Q 5126271 IC50 = 10000 nM T87831 CWA48L 5157579 IC50 = 5011.87 nM T87831 C5ZHD0 9988173 IC50 = 20 nM T87831 C80GUM 10101710 IC50 = 200 nM T87831 CDOT07 10463134 IC50 = 20 nM T87831 C8LT5E 10506680 IC50 = 600 nM T87831 C6ZDT0 10532966 IC50 = 100 nM T87831 CPXW96 10577155 IC50 = 2000 nM T87831 CEQ2K7 10579232 IC50 = 900 nM T87831 CLO6Q7 10625475 EC50 = 300 nM T87831 C2GA8T 10648894 IC50 = 2000 nM T87831 CEW7F9 10649324 IC50 = 4000 nM T87831 C4LQ2I 10696097 IC50 = 1000 nM T87831 CTXE17 10697484 EC50 = 40 nM T87831 C62TJG 10697767 EC50 = 2 nM T87831 C36INL 10700450 IC50 = 300 nM T87831 C3E5IO 10720444 IC50 = 2000 nM T87831 CR2S5U 10771672 IC50 = 500 nM T87831 C9T3ZV 10837940 IC50 = 2000 nM T87831 C7CRL9 10840230 EC50 = 900 nM T87831 CR70KN 11801040 EC50 = 1 nM T87831 CJ9NM2 14655143 IC50 = 2511.89 nM T87831 C4K5YB 24244526 IC50 = 10000 nM T87831 CIAE78 24776344 EC50 > 10000 nM T87831 C13HPO 24776345 EC50 > 10000 nM T87831 CMN49A 24776346 EC50 > 10000 nM T87831 C5GOM9 24776347 EC50 > 10000 nM T87831 CKN8F9 24776348 EC50 > 10000 nM T87831 CKXA38 24776349 EC50 > 10000 nM T87831 CUK30M 24776350 EC50 > 10000 nM T87831 C1H3PU 24776351 EC50 > 10000 nM T87831 CV26ST 24776352 EC50 > 10000 nM T87831 CGH24A 24776353 EC50 > 10000 nM T87831 CMU90L 24776354 EC50 > 10000 nM T87831 CC5LJ6 24776355 EC50 > 10000 nM T87831 C69CTS 24776356 EC50 > 10000 nM T87831 C5HVI6 24776357 EC50 > 10000 nM T87831 C90PWR 24776358 EC50 > 10000 nM T87831 C56OWF 44232675 EC50 = 2300 nM T87831 CJK72M 44232677 EC50 = 10500 nM T87831 CN74MP 44232924 EC50 = 9700 nM T87831 C2MP3Y 44232925 EC50 = 800 nM T87831 CAO83Q 44233644 EC50 = 2800 nM T87831 C3UBZ9 44233645 EC50 = 3200 nM T87831 CJ6A2K 44233646 EC50 = 1100 nM T87831 CN81VH 44233647 EC50 = 3600 nM T87831 CMY4B3 44233648 EC50 = 5700 nM T87831 CXZ1K2 44233905 EC50 = 4300 nM T87831 C8S4IJ 44236326 EC50 = 2600 nM T87831 CP2R7H 44236328 EC50 = 2238.72 nM T87831 C8KW7R 44236329 EC50 = 3900 nM T87831 CCX6A4 44236330 EC50 = 1600 nM T87831 CA5L7V 44263975 IC50 = 2000 nM T87831 CE3YW8 44263999 EC50 = 1 nM T87831 C8JKA5 47012371 IC50 = 3981.07 nM T87831 C9KDN8 54580795 EC50 = 1584.89 nM T87831 CCS14V 54580796 IC50 = 630.96 nM T87831 C1FAI5 54580798 IC50 = 1000 nM T87831 CN57AB 54581780 IC50 = 79.43 nM T87831 CM46OR 54581781 IC50 = 1584.89 nM T87831 CP9Y2R 54581782 IC50 = 5011.87 nM T87831 CMY97I 54581826 IC50 = 1995.26 nM T87831 CRU12A 54581827 IC50 = 5011.87 nM T87831 C4TV0M 54582743 IC50 = 794.33 nM T87831 C8G6CK 54582778 IC50 = 10000 nM T87831 CKL73F 54583762 IC50 = 10000 nM T87831 CSJ59H 54584752 IC50 = 3981.07 nM T87831 CVIF18 54584753 IC50 = 3162.28 nM T87831 C4UR8W 54586640 IC50 = 2511.89 nM T87831 CU7CT2 54586641 IC50 = 10000 nM T87831 C2M3ZO 54587661 IC50 = 2511.89 nM T87831 CC56RB 54587699 IC50 = 6309.57 nM T87831 C4GJQ9 54587700 IC50 > 25118.86 nM T87831 CMN1C6 54752118 IC50 = 25.12 nM T87831 C89PEN 56949822 IC50 = 3.981 nM T87831 C1K8TD 56949966 IC50 = 158.49 nM T87831 C4DOH9 57390867 IC50 = 31.62 nM T87831 C1RG5Z 57390868 IC50 = 1000 nM T87831 C2MJR7 57391103 IC50 = 6309.57 nM T87831 CA6V0T 57392729 IC50 = 3162.28 nM T87831 C41NET 57392871 IC50 = 3981.07 nM T87831 CZ1D5V 57392872 IC50 = 1584.89 nM T87831 C7G3JQ 57392882 IC50 = 316.23 nM T87831 CR3C2N 57392963 IC50 = 158.49 nM T87831 CCB3L9 57392964 IC50 = 5011.87 nM T87831 CIR50J 57394389 IC50 = 316.23 nM T87831 CY0MC7 57394598 IC50 = 10000 nM T87831 C7IJH0 57394609 IC50 = 3981.07 nM T87831 CRC3P0 57394706 IC50 = 10000 nM T87831 C04IST 57394707 IC50 = 79.43 nM T87831 C4LTG6 57394708 IC50 = 1000 nM T87831 CH7E9P 57396149 IC50 = 39.81 nM T87831 CLK5Y1 57396150 IC50 = 316.23 nM T87831 C4ZV8B 57396213 IC50 = 1000 nM T87831 C79MKF 57396214 IC50 = 398.11 nM T87831 C8DE3F 57396467 IC50 = 15848.93 nM T87831 CMHO90 57396468 IC50 = 501.19 nM T87831 CBW93G 57397970 IC50 = 10000 nM T87831 C9WIA0 57398165 IC50 = 5011.87 nM T87831 C6O0RD 57398166 IC50 = 5011.87 nM T87831 CQI64G 57398252 IC50 = 19952.62 nM T87831 C3QG1J 57398253 IC50 = 5011.87 nM T87831 C1MPH3 57398255 IC50 = 5011.87 nM T87831 CR6EN5 57398256 IC50 = 6309.57 nM T87831 CF9W1V 57398257 IC50 = 3162.28 nM T87831 CM06QZ 57398258 IC50 = 125.89 nM T87831 C6A9IL 57398259 IC50 = 1000 nM T87831 CJ09NI 57398260 IC50 = 12.59 nM T87831 CU9MV7 57399614 IC50 = 3162.28 nM T87831 C4LF8O 57399672 IC50 = 1584.89 nM T87831 C6KR9C 57399796 IC50 = 1995.26 nM T87831 C6M1QI 57399797 IC50 = 794.33 nM T87831 CN92KO 57399908 IC50 = 1584.89 nM T87831 CU2E9W 57399909 IC50 = 1000 nM T87831 C8A5MS 57399910 IC50 = 158.49 nM T87831 C8NSW3 57401368 IC50 = 199.53 nM T87831 CCS7W5 57401369 IC50 = 79.43 nM T87831 CF7JK1 57401370 IC50 = 2511.89 nM T87831 C14HAO 57401427 IC50 = 6309.57 nM T87831 CKC5S7 57401587 IC50 = 10000 nM T87831 CL6ZJ1 57401680 IC50 = 10000 nM T87831 CQ2B9I 57401681 IC50 = 79.43 nM T87831 CBG7P1 57401682 IC50 = 501.19 nM T87831 CZ7WC8 57401683 IC50 = 794.33 nM T87831 CUB6X4 57401684 IC50 = 1995.26 nM T87831 CTR5U9 57403176 IC50 = 25118.86 nM T87831 CF82EM 57403415 IC50 = 10000 nM T87831 C18MJW 57403416 IC50 = 25.12 nM T87831 CV1JC6 70691873 IC50 = 150 nM T87831 C4IEK9 71697968 IC50 = 180 nM T87831 C7YE9S 71698276 IC50 = 120 nM T87831 C67QTG 71698362 EC50 = 3000 nM T87831 CU3K2T 71698365 EC50 = 13500 nM T87831 CYT92I 71698442 EC50 = 8100 nM T87831 CK9Q5W 71698446 EC50 = 11200 nM T87831 CNI78T 71698527 EC50 = 6100 nM T87831 C25ITN 71698528 EC50 = 4200 nM T87831 C43WJT 71698529 EC50 = 4500 nM T87831 CPJ6L3 71698530 EC50 = 10800 nM T87831 CT01IM 71698531 EC50 = 9000 nM T87831 CK8V5I 71698532 EC50 > 50000 nM T87831 C5P3LQ 71698620 EC50 > 50000 nM T87831 CUI9K5 71698621 EC50 > 50000 nM T87831 CJRV63 71698622 EC50 > 50000 nM T87831 CPO3W2 71698623 EC50 > 50000 nM T87831 C05SFZ 71698624 EC50 > 50000 nM T87831 CS2TY5 71698709 EC50 > 50000 nM T87831 C7EBU6 71698710 EC50 > 50000 nM T87831 C4F5DE 71698711 EC50 > 50000 nM T87831 C6D2NC 71698712 EC50 > 50000 nM T87831 CI4FT0 71698713 EC50 > 50000 nM T87831 CW0M1S 71698793 EC50 > 50000 nM T87831 C3ALW5 71698794 EC50 > 50000 nM T87831 C27VXB 71698795 EC50 > 50000 nM T87831 C18AYL 71698796 EC50 > 50000 nM T87831 C9XQT1 71698797 EC50 > 50000 nM T87831 CH2AN3 71698877 EC50 > 50000 nM T87831 CH03IG 71698878 EC50 > 50000 nM T87831 CBTW91 71698880 EC50 = 5500 nM T87831 C7C0AG 71698881 EC50 > 50000 nM T87831 CP1FY3 71698966 EC50 = 6900 nM T87831 CU5JI8 71698967 EC50 = 6600 nM T87831 CHZ39E 71698968 EC50 = 10500 nM T87831 C9JOI7 71698969 EC50 > 50000 nM T87831 CKOY37 71698970 EC50 > 50000 nM T87831 CW7G4H 71698971 EC50 > 50000 nM T87831 C67VPX 71698972 EC50 = 5800 nM T87831 CKY03S 71699059 EC50 = 4500 nM T87831 CU13WD 71699060 EC50 = 8100 nM T87831 CM7BJ1 71699061 EC50 = 13800 nM T87831 CF92UE 71699062 EC50 = 9300 nM T87831 CPV70F 71699063 EC50 = 29300 nM T87831 C5BET3 71699064 EC50 > 50000 nM T87831 CP01IH 71699065 EC50 = 7600 nM T87831 CO03UK 71699139 EC50 = 9500 nM T87831 CQ75GP 71699140 EC50 > 50000 nM T87831 CGJ5X6 71699141 EC50 > 50000 nM T87831 CCT6F3 71699142 EC50 = 12800 nM T87831 CT81IA 71699143 EC50 = 9300 nM T87831 CYJ18T 71699222 EC50 > 50000 nM T87831 CKIS09 73345687 IC50 > 10000 nM T87831 C8E4UR 73345688 IC50 = 9200 nM T87831 CNV1O3 73346926 IC50 = 1570 nM T87831 C29SZY 73347040 IC50 = 5500 nM T87831 C53FHD 73347181 IC50 = 2300 nM T87831 C1MSA3 73347182 IC50 > 10000 nM T87831 C2GP9J 73347184 IC50 = 6330 nM T87831 CYAM67 73347185 IC50 > 10000 nM T87831 CB4Z3C 73347187 IC50 > 10000 nM T87831 CY35VS 73347188 IC50 = 3250 nM T87831 C2UMC0 73348697 IC50 = 1800 nM T87831 C8Y9BO 73348698 IC50 > 10000 nM T87831 CUV2H8 73348699 IC50 = 560 nM T87831 C02TEP 73348700 IC50 > 5000 nM T87831 CC26MI 73348702 IC50 = 590 nM T87831 C04MXE 73350273 IC50 > 10000 nM T87831 CP76MH 73350274 IC50 = 7000 nM T87831 C9YP4V 73350275 IC50 = 6300 nM T87831 C8A0FU 73350276 IC50 > 10000 nM T87831 CS50EI 73350277 IC50 = 1480 nM T87831 C4JG5S 73350278 IC50 = 2500 nM T87831 CB0ZS5 73350279 IC50 > 5000 nM T87831 CVXI38 73351612 IC50 = 6450 nM T87831 CIN06P 73351778 IC50 > 10000 nM T87831 C7SBD8 73351779 IC50 > 10000 nM T87831 CNGX73 73351780 IC50 > 10000 nM T87831 C59IQV 73351781 IC50 > 3000 nM T87831 C18FYB 73351783 IC50 > 10000 nM T87831 CGK35X 73351785 IC50 > 10000 nM T87831 CX86TP 73353255 IC50 > 10000 nM T87831 CJBS21 73353256 IC50 = 2200 nM T87831 C3WMA5 73353259 IC50 = 300 nM T87831 C57VIN 73353260 IC50 > 10000 nM T87831 CFXP14 73353261 IC50 = 570 nM T87831 C4WN9O 73354611 IC50 > 10000 nM T87831 C6LP1D 73354769 IC50 = 3400 nM T87831 CXJ53K 73354770 IC50 > 3000 nM T87831 CXD51S 73354771 IC50 > 10000 nM T87831 C29SYL 73354772 IC50 = 750 nM T87831 C0HYX7 73354773 IC50 = 3000 nM T87831 CR1T6W 73354775 IC50 > 10000 nM T87831 CAZ13T 73356299 IC50 > 3000 nM T87831 CGH64E 73356301 IC50 > 5000 nM T87831 CE4CK5 73356302 IC50 = 2520 nM T87831 CUVL53 73356305 IC50 > 10000 nM T87831 CG68MZ 92263206 IC50 = 12600 nM T87831 CODS02 102234371 IC50 = 420 nM T87831 CT3MS4 117993763 IC50 = 16500 nM T87831 CED1S3 118707168 IC50 = 140 nM T87831 CP37QL 122181231 EC50 = 260 nM T87831 C5FPZ6 122181322 EC50 = 950 nM T87831 C4Q9TF 122487956 EC50 > 100000 nM T87831 C59JDT 122487958 EC50 = 2089.3 nM T87831 C4EXO6 122487959 EC50 = 1778.28 nM T87831 CIGS34 122487963 EC50 > 100000 nM T87831 C7LN5A 122487964 EC50 = 7585.78 nM T87831 C1DFK0 122487965 EC50 = 2630.27 nM T87831 C3AF7I 122487968 EC50 = 8511.38 nM T87831 C7HY8T 122487970 EC50 = 851.14 nM T87831 CUVH13 122487971 EC50 = 1819.7 nM T87831 C93KFY 122487972 EC50 = 7943.28 nM T87831 CKO1H3 122487974 EC50 = 147.91 nM T87831 CVA02B 122487975 EC50 > 100000 nM T87831 CG3E7B 122487981 EC50 = 1230.27 nM T87831 CX71MD 122487986 EC50 = 3388.44 nM T87831 CQRU49 122487990 EC50 = 5011.87 nM T87831 CH7TR4 122488043 EC50 = 6309.57 nM T87831 CRNM14 135796853 Ki > 10000 nM T87831 CW9H4R 135796854 Ki > 10000 nM T87831 CBR72J 136118020 Ki > 10000 nM T87831 C04XKL 136118021 Ki > 10000 nM T87831 CE3G5Y 136118022 Ki > 10000 nM T87831 C4X9WU 136118023 Ki > 10000 nM T87831 CDS1T4 136118024 Ki > 10000 nM T87831 CY05OB 136118025 Ki > 10000 nM T87831 CV42NE 136118026 Ki > 10000 nM T87831 CG9DI5 136118027 Ki > 10000 nM T87831 CH1F3W 136118028 Ki > 10000 nM T87831 C87OWX 136118029 Ki > 10000 nM T87831 CV9LN3 145949892 EC50 = 1500 nM T87831 C4ON9H 145951856 EC50 = 5400 nM T87831 C1Q8YJ 145952485 EC50 = 2800 nM T87831 CRX78Z 145952664 EC50 = 10300 nM T87831 CG18UM 145953127 EC50 = 18800 nM T87831 COX71H 145954612 EC50 = 950 nM T87831 CF4M2C 145955803 EC50 = 5900 nM T87831 C2X5OV 145956276 EC50 = 630 nM T87831 CX7RA0 145956361 EC50 = 450 nM T87831 CM9C4I 145956762 EC50 = 4700 nM T87831 CN36IR 145958736 EC50 = 5200 nM T87831 CJ0B9Q 145963525 EC50 = 850 nM T87831 CU6K8I 145978177 EC50 = 2400 nM T87831 C8UY7H 146035588 EC50 = 83 nM T87831 C9S8JD 146035589 EC50 = 54.95 nM T87831 CP87OT 154706263 EC50 = 6.457 nM T87831 C6H2LN 154725143 EC50 = 331.13 nM T87831 COQ48T 155510570 IC50 = 19600 nM T87831 CK0V1N 155512026 EC50 > 100000 nM T87831 CQHD97 155514516 EC50 = 2818.38 nM T87831 C8PT1I 155516247 EC50 = 1380.38 nM T87831 C8KM2F 155517009 IC50 = 2400 nM T87831 CDXE73 155517073 IC50 = 37400 nM T87831 CC9I7T 155518804 EC50 > 100000 nM T87831 CA2LI1 155519289 EC50 = 169.82 nM T87831 C6FQE9 155519369 EC50 = 144.54 nM T87831 CB9XF8 155523344 IC50 = 540 nM T87831 C0IO5F 155523368 EC50 = 5623.41 nM T87831 C9YPK2 155523493 EC50 > 100000 nM T87831 CD63JM 155524563 IC50 = 14500 nM T87831 CR9P8T 155525710 EC50 > 100000 nM T87831 CPWN95 155526792 EC50 > 100000 nM T87831 C4F9CO 155529906 IC50 = 11700 nM T87831 C4ELN6 155535862 EC50 > 100000 nM T87831 CF8BG0 155538591 EC50 = 2630.27 nM T87831 C2KHI7 155539071 EC50 > 100000 nM T87831 C09IQU 155540456 EC50 = 1862.09 nM T87831 CMNO20 155550945 EC50 > 100000 nM T87831 CAK5L4 155553761 EC50 > 100000 nM T87831 CAQ0E6 155555363 EC50 = 6309.57 nM T87831 CX71IA 155555898 EC50 = 125.89 nM T87831 C9E8KO 155557264 EC50 > 100000 nM T87831 CADQ93 155557362 IC50 = 1080 nM T87831 CR0UM3 155558334 EC50 > 100000 nM T87831 C6JBS1 155560790 EC50 > 100000 nM T87831 C0V1ET 155561375 EC50 > 100000 nM T87831 C2L9SR 155561704 EC50 > 100000 nM T87831 CMI45H 155562717 EC50 > 100000 nM T87831 D00OMW 5322194 IC50 = 5011.87 nM T87831 D05UWQ 4329947 IC50 = 501.19 nM T87831 D09MAZ 46897162 IC50 > 5000 nM T87831 D0G5DH 53233899 IC50 = 316.23 nM T87831 D0M9RF 3092570 Ki = 100 nM T87831 D0WB8E 24776341 EC50 = 32.36 nM T87831 D0XF0A 443295 EC50 = 10 nM T94309 D0T9TJ 3034010 IC50 = 0.4 ug.mL-1 T94309 CPW9G5 65126 IC50 = 36000 nM T94309 CB4A7Z 97487 IC50 = 168600 nM T94309 CQV5G6 167963 IC50 = 17900 nM T94309 CA4K6I 278055 IC50 = 428600 nM T94309 CLV4X1 442009 IC50 = 13000 nM T94309 CG6W8R 9839754 IC50 > 10000 nM T94309 C8XQ3Z 9908564 IC50 = 120000 nM T94309 CH0R1M 10038557 IC50 > 50000 nM T94309 CEKX28 10094001 IC50 > 50000 nM T94309 CI70JE 10109540 IC50 > 10000 nM T94309 CU21VN 10476544 IC50 > 50000 nM T94309 CN3V5E 10648871 IC50 = 1.7 ug.mL-1 T94309 C0LZ5G 44445119 IC50 = 270000 nM T94309 CS98BK 44445120 IC50 = 27000 nM T94309 CN80WG 46898596 IC50 = 3200 nM T94309 C7GL0E 46898597 IC50 = 9000 nM T94309 CM9I4K 52940767 IC50 = 16000 nM T94309 CWP32U 60150482 Ki = 67000 nM T94309 C25YBT 70685571 Ki = 550000 nM T94309 CN4V8J 70685572 Ki = 170000 nM T94309 C4S7IP 70689760 Ki = 360000 nM T94309 CH4GO3 89922162 IC50 > 37000 nM T94309 C4XK0O 145949153 IC50 = 13480 nM T94309 C49FSP 145949928 IC50 = 1100 nM T94309 CX20FM 145950231 IC50 = 6900 nM T94309 CT8I2G 145952235 IC50 = 11750 nM T94309 CAVK82 145953842 IC50 = 1870 nM T94309 C3O8XZ 145955293 IC50 = 9150 nM T94309 CY1IO7 145955741 IC50 = 2280 nM T94309 CXZ24D 145958385 IC50 = 7820 nM T94309 CUF61P 145958778 IC50 = 2310 nM T94309 CFW10Z 145959167 IC50 = 14480 nM T94309 CQKN42 145959837 IC50 = 1650 nM T94309 CH6GF5 145960166 IC50 = 1250 nM T94309 CM9F5U 145960565 IC50 = 2010 nM T94309 CPW30H 145971480 IC50 = 7380 nM T95183 D0JU5X 400769 IC50 = 22000 nM T95183 CX4RD6 20176 IC50 > 5000000 nM T95183 CF2Z4P 136655 IC50 > 5000000 nM T95183 CK7M0H 290223 IC50 = 8700 nM T95183 CGV35L 2737287 IC50 > 5000000 nM T95183 C53YHR 2776547 IC50 = 1300000 nM T95183 C7MW8B 5918438 IC50 = 32560 nM T95183 CT0O5K 10634145 IC50 > 31600 nM T95183 C5IY6B 17254167 IC50 = 3300 nM T95183 CMOK20 17399295 IC50 > 100000 nM T95183 CYA13H 45352259 IC50 > 50000 nM T95183 CEU7P1 86276129 IC50 > 100000 nM T95183 CIFM91 137642808 IC50 = 66080 nM T95183 CE1BG8 155526632 IC50 = 9700 nM T44282 D01WGJ 107971 IC50 = 40 nM T44282 CP49EN 15134 IC50 = 229.33 nM T44282 CBKM24 54357 IC50 = 2100 nM T44282 CVG38C 67114 IC50 < 15000 nM T44282 CDL3E1 262696 IC50 > 100000 nM T44282 C2XYO5 442813 IC50 > 6000 nM T44282 C7JT8K 611621 Ki = 1000 nM T44282 C4X2YG 666267 IC50 > 100000 nM T44282 CPG42Y 666623 IC50 > 100000 nM T44282 C4IP8H 707701 IC50 = 360 nM T44282 C9WAT8 707707 Ki = 35 nM T44282 CI8C6S 707714 IC50 = 67 nM T44282 CNWH76 707732 IC50 = 340 nM T44282 C5VU7F 707801 IC50 = 150 nM T44282 C2TK3I 854708 IC50 = 67 nM T44282 CJ1CV6 906688 IC50 = 150 nM T44282 C32WDZ 1581092 IC50 = 1700 nM T44282 C6H8JE 1633306 Ki = 5600 nM T44282 CP1QI9 1894707 IC50 = 3500 nM T44282 CM16ZY 1912440 IC50 > 100000 nM T44282 CGJ84F 1966642 IC50 > 100000 nM T44282 C8VWZ5 2057118 IC50 > 100000 nM T44282 CMCI42 2166081 IC50 > 100000 nM T44282 COW7J9 2265401 IC50 = 50 nM T44282 CXG6M7 2282752 IC50 = 1200 nM T44282 C6ZTD4 2296065 IC50 > 100000 nM T44282 C9AR5J 2902827 IC50 = 1500 nM T44282 CNH4Q5 2930041 IC50 = 410 nM T44282 CTM42Y 3062796 IC50 = 2500 nM T44282 CEQ0V8 3586132 Ki = 19 nM T44282 CP7G8W 3596579 IC50 = 260 nM T44282 CQ0AR8 3704739 IC50 = 2100 nM T44282 CL59PA 3782756 Ki = 310 nM T44282 CW63PI 4118326 IC50 = 400 nM T44282 C5ENU0 4165008 IC50 = 150 nM T44282 C5K7QS 4198873 IC50 = 40 nM T44282 C79OMC 4653534 IC50 > 100000 nM T44282 CZY6A7 4914255 Ki = 1100 nM T44282 C09QCN 4999777 IC50 > 100000 nM T44282 C5LGJ1 5282362 IC50 = 7000 nM T44282 CO0D3B 6954241 Ki = 2400 nM T44282 C8MD5K 9797371 IC50 = 250 nM T44282 C2PLU8 9819934 IC50 = 100 nM T44282 C43XWS 9843294 IC50 = 270 nM T44282 CP25HN 9867778 IC50 = 3 nM T44282 CUX4A2 9885593 IC50 = 9 nM T44282 CGK1S3 9888593 IC50 = 50 nM T44282 C8CWV9 9907990 IC50 = 9 nM T44282 C85ICB 9998250 IC50 = 100 nM T44282 C39IDW 10193224 IC50 = 1200 nM T44282 C2HN1O 10384506 IC50 >> 9000 nM T44282 CC51PD 10432095 IC50 = 300 nM T44282 C08RKO 10475227 IC50 = 40 nM T44282 CD7N1Y 10613705 IC50 = 800 nM T44282 CP2YR9 10687704 IC50 = 100 nM T44282 C12CSD 10862798 IC50 = 7200 nM T44282 CDY3M9 10904674 IC50 = 1000 nM T44282 CVM8Z6 10914713 IC50 = 1500 nM T44282 C1OYA8 10916836 IC50 > 9000 nM T44282 CG1P0O 10925737 IC50 = 150 nM T44282 C6RME5 10926283 IC50 = 120 nM T44282 CS2H7X 10949302 IC50 = 40 nM T44282 C9XCR6 10958746 IC50 = 130 nM T44282 CKV9C4 11002709 IC50 = 320 nM T44282 C1OZ7J 11037528 IC50 = 1700 nM T44282 CMV68C 11090565 IC50 = 700 nM T44282 CYXG05 11143753 IC50 = 2000 nM T44282 CUQ1L4 11728663 IC50 = 240 nM T44282 C7Z1VD 11732018 IC50 = 280 nM T44282 C3M6TY 11733922 IC50 > 9000 nM T44282 CBGA07 11748522 IC50 = 70 nM T44282 C4E0QO 11761097 IC50 = 4500 nM T44282 CVT56D 11762178 IC50 = 130 nM T44282 CN8QJ5 13165000 IC50 = 470 nM T44282 CQH86P 28492659 IC50 = 100 nM T44282 CG6XI0 44340754 IC50 = 3500 nM T44282 CX9P7I 142581415 IC50 = 5000 nM T44282 CEHC09 142581553 IC50 = 5000 nM T44282 D0A9RM 5281804 Ki = 450 nM T44282 D0O0LU 264734 Ki = 15000 nM T44282 D0O9UY 10469827 IC50 = 80 nM T44282 D0OC4B 5357479 IC50 = 1500 nM T44282 D0SY2M 5281708 IC50 = 9000 nM T91390 C12MJF 5281098 IC50 = 296 nM T91390 CX9L4Y 127043462 IC50 = 94.5 nM T91390 CR7QK2 127043679 IC50 = 1.9 nM T91390 C79PSH 127044134 IC50 = 4.07 nM T91390 C3B0RE 127044297 IC50 > 10000 nM T91390 C4S0PV 127044320 IC50 > 1250 nM T91390 C8NJB0 127044321 IC50 > 10000 nM T91390 CQ9FT5 127044322 IC50 > 20000 nM T91390 CYG35R 127044323 IC50 > 20000 nM T91390 CGJ72V 127044324 IC50 > 20000 nM T91390 C34EOL 127044325 IC50 = 1.3 nM T91390 CHGM40 127044326 IC50 = 12.8 nM T91390 CUDO70 127044327 IC50 = 12.2 nM T91390 C64ITM 127044642 IC50 > 2500 nM T91390 CS52JP 127044643 IC50 > 10000 nM T91390 CVR92K 127044644 IC50 > 10000 nM T91390 CR2P6L 127044645 IC50 > 10000 nM T91390 C8H4WN 127044646 IC50 = 12.2 nM T91390 CRE2O4 127044812 IC50 > 1250 nM T91390 C1UZ8M 127044970 IC50 > 10000 nM T91390 CM0QS2 127044971 IC50 = 808.3 nM T91390 C1TO9Y 127044972 IC50 = 603.1 nM T91390 C4OEW8 127044973 IC50 = 201.9 nM T91390 CCV5I6 127044980 IC50 = 8.8 nM T91390 CX7DH4 127044981 IC50 = 12.4 nM T91390 C6P1NL 127045116 IC50 > 2500 nM T91390 CP5Q8K 127045117 IC50 > 1000 nM T91390 CY92VX 127045118 IC50 = 31 nM T91390 CT83QE 127045119 IC50 = 39.4 nM T91390 CM1Q8D 127045120 IC50 = 7.8 nM T91390 CD8X3H 127045124 IC50 = 10 nM T91390 CI80BD 127045125 IC50 > 5000 nM T91390 CW95UD 127045126 IC50 = 245.6 nM T91390 CKA84F 127045127 IC50 = 770.1 nM T91390 C8D0NA 127045128 IC50 > 1000 nM T91390 CYC70B 127045129 IC50 > 50000 nM T91390 CK1S0N 127045574 IC50 > 10000 nM T91390 C8WT5A 127048974 IC50 = 219 nM T91390 C78DQY 127050268 IC50 = 683.7 nM T91390 C05ILG 127050578 IC50 = 740.2 nM T91390 C3I0UD 127051173 IC50 = 355.1 nM T91390 C35JLQ 127051177 IC50 = 300 nM T91390 C73JKV 137631429 IC50 > 1000 nM T91390 C7K9BV 137631433 IC50 > 1000 nM T91390 CGNH80 137631598 IC50 = 62.8 nM T91390 CBY4W9 137631701 IC50 = 27.3 nM T91390 C5H0JC 137632052 IC50 = 7.7 nM T91390 C9P5GJ 137632416 IC50 = 400.4 nM T91390 CDA47Y 137632623 IC50 = 9.5 nM T91390 CLE85P 137632936 IC50 = 256.5 nM T91390 CTR4O2 137633026 IC50 > 1000 nM T91390 CWF8K5 137633093 IC50 = 700 nM T91390 CWY2I4 137633238 IC50 > 1000 nM T91390 CW1SF5 137633301 IC50 > 1000 nM T91390 C05ILH 137633336 IC50 = 4.7 nM T91390 CGJN45 137633438 IC50 > 1000 nM T91390 C4HE2R 137633726 IC50 > 1000 nM T91390 CQJ6H2 137633967 IC50 > 1000 nM T91390 C1PWI8 137634054 IC50 > 1000 nM T91390 C53TNY 137634407 IC50 > 1000 nM T91390 C9GB7R 137634482 IC50 = 43.5 nM T91390 CLTX83 137634586 IC50 = 2.5 nM T91390 CJRB52 137634605 IC50 > 1000 nM T91390 C2T8RL 137634909 IC50 > 1000 nM T91390 CBJ17S 137634915 IC50 > 1000 nM T91390 CM1ZP9 137635056 IC50 = 83.8 nM T91390 CX7GA4 137635351 IC50 = 3.8 nM T91390 CLF90K 137635683 IC50 > 1000 nM T91390 C53NOY 137635836 IC50 > 1000 nM T91390 CMB9N4 137636070 IC50 > 1000 nM T91390 CO3BL0 137636178 IC50 > 1000 nM T91390 C7J0CW 137636181 IC50 > 1000 nM T91390 CC0OH5 137636293 IC50 = 131.8 nM T91390 C7AEV5 137636300 IC50 > 1000 nM T91390 CLAX45 137636307 IC50 > 1000 nM T91390 C6M9AG 137636471 IC50 = 33.5 nM T91390 CKH1R0 137636972 IC50 = 15.8 nM T91390 C0CXO1 137637098 IC50 = 463.6 nM T91390 CX5IZ0 137637109 IC50 = 23.5 nM T91390 CG27UX 137637163 IC50 = 238.6 nM T91390 CD1XT2 137637349 IC50 > 1000 nM T91390 CS6W3J 137637456 IC50 > 1000 nM T91390 C3E1IR 137637523 IC50 = 253.6 nM T91390 C9XZ2R 137637785 IC50 = 91.3 nM T91390 C7JGL9 137638222 IC50 = 167 nM T91390 CL3VO9 137638249 IC50 > 1000 nM T91390 C3Y4BT 137638332 IC50 = 54.4 nM T91390 CH5F7N 137638539 IC50 > 1000 nM T91390 CC09VU 137638599 IC50 = 4.8 nM T91390 CP3TF4 137639291 IC50 > 1000 nM T91390 C5KI0S 137639580 IC50 > 1000 nM T91390 C31OHQ 137639762 IC50 > 1000 nM T91390 C4DW9S 137639931 IC50 = 4.5 nM T91390 C4K6QZ 137640078 IC50 > 1000 nM T91390 CU26TA 137640577 IC50 > 1000 nM T91390 CXG26Z 137640751 IC50 = 142.6 nM T91390 CZW7J9 137640880 IC50 > 1000 nM T91390 CA60UH 137640930 IC50 = 279.6 nM T91390 C91TKH 137640933 IC50 > 1000 nM T91390 CUX26G 137640990 IC50 > 1000 nM T91390 C01UFJ 137641337 IC50 > 1000 nM T91390 C1XWO4 137641464 IC50 = 642.4 nM T91390 CQ47EZ 137641569 IC50 > 1000 nM T91390 CR86NX 137641816 IC50 = 6.2 nM T91390 CK9OV0 137641833 IC50 = 12.3 nM T91390 CH4QU8 137641902 IC50 > 1000 nM T91390 C1X4YC 137642015 IC50 > 1000 nM T91390 CEO1L5 137642193 IC50 > 1000 nM T91390 CH79XT 137642505 IC50 = 17.3 nM T91390 CIX8G0 137642672 IC50 > 1000 nM T91390 C4N7MQ 137642784 IC50 > 1000 nM T91390 CYWA72 137643103 IC50 = 6.5 nM T91390 C2W3MP 137643125 IC50 > 1000 nM T91390 C58ISN 137643139 IC50 = 400 nM T91390 CKX9Y8 137643477 IC50 = 89.6 nM T91390 CW84CS 137643538 IC50 > 1000 nM T91390 CU17NV 137643725 IC50 = 784.7 nM T91390 CG3A9D 137643738 IC50 > 1000 nM T91390 CB1T9O 137643828 IC50 > 1000 nM T91390 CL3V2D 137644044 IC50 = 199 nM T91390 CP1JC4 137644431 IC50 > 1000 nM T91390 C0EDP1 137644453 IC50 = 6.4 nM T91390 C0ONB9 137644544 IC50 > 1000 nM T91390 CHS17L 137644882 IC50 = 5.2 nM T91390 C1Z7NM 137644951 IC50 > 1000 nM T91390 C3UCS8 137645305 IC50 = 101.8 nM T91390 CGI58R 137645414 IC50 = 74.1 nM T91390 CAV69W 137645467 IC50 > 1000 nM T91390 C0SGD6 137645492 IC50 > 1000 nM T91390 CP1ST3 137645812 IC50 > 1000 nM T91390 CVF1L0 137646006 IC50 = 73.1 nM T91390 C4B2AS 137646232 IC50 > 1000 nM T91390 C3ATV6 137646312 IC50 = 9.9 nM T91390 C2JMQ4 137646587 IC50 = 17.8 nM T91390 C4JC2T 137646951 IC50 = 6.4 nM T91390 CCW02A 137646984 IC50 = 43.4 nM T91390 CUM6J2 137647093 IC50 > 1000 nM T91390 CDM5F8 137647124 IC50 > 1000 nM T91390 CG9U3X 137647321 IC50 = 5.9 nM T91390 CNR8K4 137647433 IC50 > 1000 nM T91390 CDN69P 137647759 IC50 > 1000 nM T91390 CS27DE 137648062 IC50 > 1000 nM T91390 CCWK52 137648217 IC50 > 1000 nM T91390 C84GQJ 137648232 IC50 = 86.4 nM T91390 C6W8NL 137648448 IC50 = 49 nM T91390 C10ZDO 137648467 IC50 = 73.2 nM T91390 C2V9SY 137649176 IC50 = 50.2 nM T91390 C7SXI2 137649457 IC50 = 2.2 nM T91390 CM2T6V 137649523 IC50 > 1000 nM T91390 CLE83H 137649637 IC50 > 1000 nM T91390 CO9AB4 137649673 IC50 = 102.1 nM T91390 C6TV5S 137649887 IC50 > 1000 nM T91390 C9L1IT 137649947 IC50 > 1000 nM T91390 CHEO50 137649974 IC50 > 1000 nM T91390 C91BTQ 137649988 IC50 > 1000 nM T91390 CP6F7W 137650046 IC50 = 3 nM T91390 CI7F1J 137650316 IC50 = 5.2 nM T91390 CX34AI 137650411 IC50 > 1000 nM T91390 CGCO94 137650575 IC50 > 1000 nM T91390 CH90XP 137650962 IC50 > 1000 nM T91390 CAQS13 137651002 IC50 > 1000 nM T91390 CCB46U 137651234 IC50 > 1000 nM T91390 CXM7C1 137651346 IC50 > 1000 nM T91390 CYN50O 137651349 IC50 > 1000 nM T91390 C6TPI4 137651640 IC50 > 1000 nM T91390 CH45NU 137651693 IC50 > 1000 nM T91390 C2GX0K 137651775 IC50 > 1000 nM T91390 CMO69Q 137652003 IC50 > 1000 nM T91390 CS9O5T 137652037 IC50 = 87.8 nM T91390 C5U4DB 137652299 IC50 = 16 nM T91390 CU2K6P 137652334 IC50 = 12.4 nM T91390 C3KDX9 137652617 IC50 = 24.5 nM T91390 CBAE35 137652679 IC50 > 1000 nM T91390 CSYA85 137652691 IC50 > 1000 nM T91390 C0OA7W 137652788 IC50 = 6.9 nM T91390 CPNG41 137653155 IC50 > 1000 nM T91390 C5GAR0 137653351 IC50 > 1000 nM T91390 CH5I1G 137653356 IC50 > 1000 nM T91390 CD1C5I 137653384 IC50 > 1000 nM T91390 C01MQU 137653509 IC50 > 1000 nM T91390 CPI13A 137653513 IC50 = 397.3 nM T91390 C0QZ1Y 137653747 IC50 = 654.4 nM T91390 C4AQS0 137653772 IC50 = 4.6 nM T91390 CVBC79 137653856 IC50 = 2.1 nM T91390 CSZQ39 137653987 IC50 > 1000 nM T91390 C2OR5W 137654018 IC50 > 1000 nM T91390 CW6M2Y 137654428 IC50 > 1000 nM T91390 C46DKN 137654445 IC50 = 8.7 nM T91390 CTE02I 137654452 IC50 = 9.5 nM T91390 CAH0J9 137654474 IC50 > 1000 nM T91390 CY4P5A 137654583 IC50 > 1000 nM T91390 CL3VY7 137654760 IC50 > 1000 nM T91390 CI0BY3 137654895 IC50 > 1000 nM T91390 C2GQ9S 137654897 IC50 > 1000 nM T91390 C9VAL5 137654958 IC50 = 20.4 nM T91390 C4ZY3D 137655037 IC50 > 1000 nM T91390 COV8G9 137655240 IC50 > 1000 nM T91390 CBNZ31 137655361 IC50 > 1000 nM T91390 C6U4VR 137655635 IC50 = 29 nM T91390 CTYK29 137656220 IC50 = 64.3 nM T91390 CL5JG9 137656440 IC50 > 1000 nM T91390 COHS03 137656666 IC50 > 1000 nM T91390 C8JW6P 137656767 IC50 > 1000 nM T91390 CQU64J 137656881 IC50 = 9.8 nM T91390 C6IVU4 137657229 IC50 > 1000 nM T91390 C6C7FX 137657428 IC50 = 5.8 nM T91390 C1SAF3 137657617 IC50 > 1000 nM T91390 CLS81C 137657723 IC50 = 9.9 nM T91390 CQGY82 137657879 IC50 = 359.8 nM T91390 CB7C5E 137657969 IC50 = 5.9 nM T91390 CHOI17 137658113 IC50 = 141.6 nM T91390 C0TC8Q 137658440 IC50 > 1000 nM T91390 C8DG0J 137658467 IC50 > 1000 nM T91390 C1PAE5 137658667 IC50 > 1000 nM T91390 C0HQI2 137658868 IC50 = 4.9 nM T91390 C1Q7BK 137658908 IC50 = 48.4 nM T91390 CWR5S8 137658999 IC50 > 1000 nM T91390 CH9W7X 137659002 IC50 = 9.2 nM T91390 CM8D0K 137659115 IC50 > 1000 nM T91390 CE2W5B 137659263 IC50 > 1000 nM T91390 CR21FL 137659613 IC50 > 1000 nM T91390 C9E0VF 137659964 IC50 = 64.8 nM T91390 CVR64W 137660114 IC50 > 1000 nM T91390 CCJP09 137660269 IC50 > 1000 nM T91390 CG9R5Z 137660325 IC50 = 74.1 nM T91390 C6GN8Z 137660334 IC50 = 5.2 nM T91390 CH1YF0 137660403 IC50 = 19.4 nM T91390 C8T0RM 137660728 IC50 > 1000 nM T91390 C5O4EK 137660774 IC50 = 80.1 nM T91390 C9QHV0 137660822 IC50 = 200 nM T91390 CAJ03K 137661265 IC50 = 564.6 nM T91390 CW48IN 137661342 IC50 > 1000 nM T91390 C5BUJ4 137662051 IC50 = 9 nM T91390 CU59VJ 137662131 IC50 = 117.9 nM T91390 CLC41T 145957467 IC50 = 430 nM T91390 CILC62 145957718 IC50 = 407.8 nM T91390 COME29 145978926 IC50 = 111.6 nM T91390 CK68MV 145979153 IC50 = 8.2 nM T91390 CDX18B 145979294 IC50 > 1000 nM T91390 C2ODH5 145980303 IC50 = 227.7 nM T91390 CN31ER 145980389 IC50 > 1000 nM T91390 C08UZQ 145980633 IC50 = 370.9 nM T91390 CCUX32 145980634 IC50 = 220.6 nM T91390 CU30NK 145980810 IC50 = 43.4 nM T91390 C3KV7L 145980833 IC50 = 8.2 nM T91390 CWMG38 145980998 IC50 > 1000 nM T91390 CG58FX 145981188 IC50 > 1000 nM T91390 C50JFC 145981269 IC50 = 15 nM T91390 C0QWN2 145981606 IC50 = 1.1 nM T91390 CLB76D 145981884 IC50 > 1000 nM T91390 C48ASI 145982063 IC50 > 1000 nM T91390 C6LIA3 145982122 IC50 = 48.6 nM T91390 CM7KC6 145982468 IC50 > 1000 nM T91390 C47GQI 145984405 IC50 > 1000 nM T91390 CVY94N 145984901 IC50 > 1000 nM T91390 CP59MN 145986781 IC50 = 8.8 nM T91390 CZV2X4 145987321 IC50 = 156 nM T91390 CRC8A2 145987463 IC50 = 19.2 nM T91390 CL2Y9Q 145987865 IC50 = 6.7 nM T91390 CR6VM4 145988576 IC50 > 1000 nM T91390 CQ37CE 145988636 IC50 = 18.9 nM T91390 CB26RW 145988860 IC50 = 20.1 nM T91390 C8Y9AP 145989328 IC50 = 4.1 nM T91390 C4EB6Y 145989887 IC50 = 43.5 nM T91390 CH5KI1 145991195 IC50 = 3.2 nM T91390 C9WU5F 145991707 IC50 = 0.4 nM T91390 CD2GA9 145991999 IC50 = 57.9 nM T91390 CN89ME 145992682 IC50 = 90.3 nM T91390 CX2ZW7 145992851 IC50 > 1000 nM T91390 C91EUQ 145993184 IC50 = 0.6 nM T91390 CI7W9Z 145993481 IC50 > 1000 nM T91390 CT4KM8 145993703 IC50 = 320.8 nM T91390 CLD92J 145994145 IC50 = 13.7 nM T78198 D06IAR 60961 Ki = 2000000 nM T78198 D0B5MP 135398513 Ki = 91000 nM T78198 D02ZKR 135449518 Ki = 0.0085 nM T78198 D02ZUO 135409409 Ki = 0.056 nM T78198 D04CWI 10445549 Ki = 33 nM T78198 D08NKJ 135398634 Ki = 5000 nM T78198 D08OBT 135413525 Ki = 13.5 nM T78198 D05UPB 135418360 Ki = 830 nM T78198 CP4C0N 55710 IC50 = 77000 nM T78198 C7TAD0 124316 IC50 > 300000 nM T78198 C7TH6K 126493 IC50 = 42600 nM T78198 CWE74G 126915 Ki = 1680000 nM T78198 CV0M6A 128388 IC50 = 9900 nM T78198 CA4TO0 147047 IC50 = 142500 nM T78198 CHF50L 250702 IC50 = 112000 nM T78198 C7SRI1 260064 Ki = 550000 nM T78198 CO3U7N 493146 Ki = 580000 nM T78198 C8TL5B 493147 Ki = 780000 nM T78198 C0C8FJ 493148 Ki = 520000 nM T78198 C8KRJ3 493149 Ki = 1480000 nM T78198 CV8R5P 493150 Ki = 100000 nM T78198 C6SKA0 493151 Ki = 2210000 nM T78198 CL41IC 493152 Ki = 560000 nM T78198 C17XES 493153 Ki = 300000 nM T78198 CP3IS6 493154 Ki = 350000 nM T78198 C0D9MX 2033102 IC50 = 13400 nM T78198 CW43RI 15741979 IC50 = 95000 nM T78198 CA5U0D 15741991 IC50 = 11400 nM T78198 CU2JW8 15741996 IC50 > 75000 nM T78198 C50PLT 15741997 IC50 > 150000 nM T78198 CZ4LC9 15741998 IC50 = 5000 nM T78198 C34MPO 15742001 IC50 = 4600 nM T78198 CD9H5W 15742002 IC50 = 5200 nM T78198 C1E3QW 15742003 IC50 = 8900 nM T78198 CQ1Y9G 44264323 Ki = 1400 nM T78198 CIFW25 44282426 IC50 = 131000 nM T78198 C0D4ES 44287558 Ki = 0.096 nM T78198 C6X9QM 44341326 Ki = 30000 nM T78198 CU73FM 44341905 Ki = 10000 nM T78198 CH0DT2 44342612 Ki > 30000 nM T78198 C7Q6PY 44342665 Ki = 4.7 nM T78198 C5U4OJ 44342899 Ki = 24.7 nM T78198 CTF16R 46233579 IC50 = 300000 nM T78198 CB2CY9 46233580 IC50 = 315000 nM T78198 CRVK79 46875976 Ki = 80000 nM T78198 C8HLD6 46876001 Ki = 20000 nM T78198 C50ZDM 90663688 Ki = 100000 nM T78198 CM8C0N 90663690 Ki > 300000 nM T78198 CG6F5Q 135400900 IC50 = 1600 nM T78198 C8WOK9 135400908 Ki = 67 nM T78198 CY4F7E 135404917 Ki = 3.7 nM T78198 CM39DW 135407110 Ki = 1800000 nM T78198 CSE1H8 135407786 Ki = 9 nM T78198 CHW8F3 135410228 IC50 = 250 nM T78198 C3YO0I 135410327 Ki = 0.0028 nM T78198 CRQ9T5 135410344 Ki = 170 nM T78198 CL46SA 135416133 IC50 = 29600 nM T78198 CV2KX1 135417285 Ki = 65 nM T78198 C94ISH 135418361 Ki = 830 nM T78198 CL1TD3 135419248 Ki = 550 nM T78198 CO52WX 135419353 Ki = 13 nM T78198 CHL2S1 135424596 IC50 = 57 nM T78198 CT6GV4 135428105 Ki = 1.26 nM T78198 CHF87B 135430577 Ki = 49 nM T78198 CS5ZR8 135433598 IC50 = 51 nM T78198 CP4EL0 135433982 Ki = 15.2 nM T78198 C7A1ZB 135434008 Ki = 3.1 nM T78198 CY82FU 135434163 Ki = 4.2 nM T78198 C3EMF2 135439532 Ki = 360 nM T78198 CC7R4J 135453934 Ki = 10000 nM T78198 C3XKO0 135457481 Ki = 10 nM T78198 C8QJT3 135457965 IC50 = 20 nM T78198 C5TA2H 135461783 Ki = 56 nM T78198 CCWR24 135461796 Ki = 530 nM T78198 CS6TZ3 135462241 Ki = 230 nM T78198 C3O0MR 135464138 Ki = 48 nM T78198 C5GER3 135464166 IC50 = 31 nM T78198 CYA6C7 135464196 IC50 = 300 nM T78198 C1MH3N 135465571 Ki = 23000 nM T78198 CDY51K 135467717 Ki = 580 nM T78198 CT4JV2 135467788 Ki = 1000 nM T78198 C0FBS9 135469331 Ki = 13400 nM T78198 CC74WR 135471400 Ki = 7300 nM T78198 CKD1P0 135480682 Ki = 18700 nM T78198 C98HEV 135484581 Ki = 100 nM T78198 C6RZE7 135487459 Ki = 0.38 nM T78198 C2GV1P 135493492 Ki = 1100 nM T78198 C1RP2D 135494321 Ki = 3.2 nM T78198 CH6QG5 135494363 Ki = 1.1 nM T78198 C9F4TM 135496257 IC50 = 47 nM T78198 CZ32JF 135496402 Ki = 220 nM T78198 C20FGO 135499988 Ki = 8.8 nM T78198 C5OV0S 135503813 Ki = 160 nM T78198 CSL8T1 135509403 Ki = 0.104 nM T78198 C49BED 135512468 Ki = 60 nM T78198 CC5M4D 135513747 Ki = 190 nM T78198 CQ9H0T 135513930 Ki = 390 nM T78198 C47QKY 135513959 Ki = 1.8 nM T78198 CR7OD9 135516802 Ki = 51 nM T78198 CT3X0N 135517351 Ki = 57 nM T78198 CT4G8Z 135517420 Ki = 1100 nM T78198 C05ZQR 135524571 Ki = 15000 nM T78198 CIZ69U 135528724 Ki = 1600 nM T78198 C8FBI4 135529765 Ki = 96 nM T78198 CJFP31 135529934 Ki = 1.3 nM T78198 C3RW8B 135535924 Ki = 12400 nM T78198 C2E6WR 135536690 IC50 = 270 nM T78198 CY49NW 135537118 IC50 = 300000 nM T78198 CTBP07 135541915 Ki = 306.1 nM T78198 CWF41T 135541926 Ki = 1 nM T78198 CN9AD0 135552935 IC50 = 23 nM T78198 CS3EZ9 135552936 IC50 = 100 nM T78198 C0XYO3 135554423 IC50 = 29.6 nM T78198 CV9LR1 135554446 IC50 ~ 330000 nM T78198 CMNH16 135566455 Ki = 1 nM T78198 CK3A4M 135566506 Ki = 0.0086 nM T78198 C6GYN0 135567191 Ki = 1100 nM T78198 CA4XW3 135678234 Ki = 270000 nM T78198 CCD02B 135678236 Ki = 3500 nM T78198 C0K4YA 135678238 Ki = 8.3 nM T78198 C6NUH3 135678240 Ki = 5.8 nM T78198 C9CA6U 135678242 Ki = 69 nM T78198 CRO54V 135678244 Ki = 60 nM T78198 CU9AJ7 135678246 Ki = 13 nM T78198 C2PB0E 135723753 Ki = 0.62 nM T78198 C97TES 135723754 Ki = 0.21 nM T78198 CL70TR 135723755 Ki = 14.9 nM T78198 CTIP20 135723756 Ki = 96 nM T78198 CC43WX 135723757 Ki = 165 nM T78198 C97MQF 135723758 Ki = 0.0052 nM T78198 CR07SK 135723759 Ki = 0.43 nM T78198 C0ZEI9 135723761 Ki = 4.3 nM T78198 CIU73Q 135723767 Ki = 4.2 nM T78198 C5IMR3 135723770 Ki = 1 nM T78198 CNU4L5 135723771 Ki = 5.2 nM T78198 C42IHU 135723892 IC50 = 11 nM T78198 C3O6EZ 135723893 IC50 = 17.9 nM T78198 CQWS23 135723894 IC50 = 11 nM T78198 CDZ28N 135726991 IC50 = 13 nM T78198 CL37WR 135726992 IC50 = 11 nM T78198 CI6V8E 135726993 IC50 = 200 nM T78198 CL85NO 135726994 IC50 = 23 nM T78198 C0O9DT 135726995 IC50 = 97 nM T78198 CEW98L 135776352 IC50 = 31400 nM T78198 CEUH36 135776353 IC50 = 5400 nM T78198 C4QD8O 135778774 Ki = 150 nM T78198 CD76PZ 135778776 Ki = 600 nM T78198 CN3V2L 135783310 Ki = 0.229 nM T78198 CTEL89 135783311 Ki = 6.3 nM T78198 C58DFV 135783313 Ki = 280 nM T78198 C3BCW7 135783314 Ki = 0.26 nM T78198 C8MD6V 135789843 IC50 = 1000 nM T78198 CX6EH7 135815064 IC50 = 47.6 nM T78198 COI9F0 135858780 Ki = 0.0021 nM T78198 CW9XE1 135858782 Ki = 0.469 nM T78198 CIV6D9 135858784 Ki = 7.5 nM T78198 C1EZ2B 135858786 Ki = 0.0086 nM T78198 C13ZUH 135858789 Ki = 0.78 nM T78198 C7IU3X 135858794 Ki = 300 nM T78198 COG59I 135858795 Ki = 31 nM T78198 CF21UL 135858821 Ki = 1.1 nM T78198 CA5JK3 135858823 Ki = 25 nM T78198 C76CKI 135873095 IC50 = 173 nM T78198 CBI9T1 135875971 Ki = 12.9 nM T78198 CP32IK 135886360 Ki = 0.032 nM T78198 CWG5P8 135900252 Ki = 1.82 nM T78198 CDO15N 135914684 Ki = 227 nM T78198 C2ASJ6 135914706 Ki = 900 nM T78198 CDL6V4 135914708 Ki = 14.1 nM T78198 CS8TF7 135914710 Ki = 3.7 nM T78198 C6RL9D 135950209 IC50 = 100 nM T78198 CRH6F8 135950240 Ki = 3.5 nM T78198 C2EW4O 135957050 Ki = 5.3 nM T78198 C0KA8P 135965877 IC50 = 100 nM T78198 C3SL1Z 135965989 IC50 = 100 nM T78198 C1HW8O 135966076 IC50 = 100 nM T78198 CIX62R 135974130 Ki = 35 nM T78198 CFZV85 135976350 Ki = 176 nM T78198 CSJT51 135976351 Ki = 200 nM T78198 C9VUF5 135976353 Ki = 37000 nM T78198 CAU40E 135976354 Ki = 7000 nM T78198 CWJ15O 135976355 Ki = 93000 nM T78198 C9MJ6F 135976360 Ki = 26000 nM T78198 CI80FP 135976361 Ki = 450 nM T78198 C4FAM6 135981941 Ki = 0.0019 nM T78198 CQ0M7E 135981944 Ki = 84 nM T78198 CSU50B 135981977 Ki = 1.4 nM T78198 CH06VS 135999964 Ki = 12700 nM T78198 CFM0K3 135999965 Ki = 0.0068 nM T78198 CAYF50 135999969 Ki = 2.84 nM T78198 CJU34V 136008868 Ki = 84 nM T78198 CU28IS 136016335 Ki = 2 nM T78198 CA4P3G 136016336 Ki = 316.3 nM T78198 CG76RC 136016337 Ki = 306.1 nM T78198 CF18TI 136016338 Ki = 30.6 nM T78198 CRO60J 136016339 Ki = 112.2 nM T78198 C9I8UL 136016340 Ki = 2.5 nM T78198 CZL19M 136016341 Ki = 10.2 nM T78198 CXH04P 136016342 Ki = 2040.8 nM T78198 CR0S3A 136020074 Ki = 16 nM T78198 C9X3JN 136020077 Ki = 6 nM T78198 CM7Y8W 136029171 Ki = 2 nM T78198 CJD2A4 136035258 IC50 = 37 nM T78198 C2XPK7 136035259 Ki = 28.2 nM T78198 CKY8L1 136036204 Ki = 0.0034 nM T78198 C52MUD 136036205 Ki = 0.4 nM T78198 CU73KB 136036206 Ki = 0.78 nM T78198 CC06TS 136036207 Ki = 1.3 nM T78198 CNT69R 136036208 Ki = 1.3 nM T78198 CENY68 136036209 Ki = 190 nM T78198 CL97TV 136054568 IC50 = 80000 nM T78198 CSLH68 136054570 IC50 = 12500 nM T78198 CVU2X7 136054571 IC50 = 25 nM T78198 C8XU2M 136055830 IC50 = 0.47 nM T78198 CP3IL7 136055831 IC50 = 0.25 nM T78198 C0VMK5 136055835 IC50 = 21.9 nM T78198 CH53CS 136055844 IC50 = 4.05 nM T78198 COCH28 136055847 IC50 = 0.085 nM T78198 CL53YX 136055848 IC50 = 0.16 nM T78198 CJ80ZM 136059690 Ki = 1.1 nM T78198 C79XUH 136066046 IC50 = 170 nM T78198 CJRY36 136066048 Ki = 5.3 nM T78198 C18ECU 136066049 Ki = 13 nM T78198 C2HF7O 136066050 Ki = 5.6 nM T78198 CV7TJ9 136074289 IC50 = 900 nM T78198 CTE1Q7 136074301 Ki = 110000 nM T78198 CI8SO1 136074302 Ki = 7000 nM T78198 C9VRK0 136076371 Ki = 10.1 nM T78198 C3BU6Z 136076372 Ki = 7 nM T78198 CEB20N 136076373 Ki = 25 nM T78198 CTA1D4 136087121 Ki = 210 nM T78198 CA4I7J 136114660 Ki = 630 nM T78198 C86CWB 136131578 Ki = 0.39 nM T78198 CE4T9N 136131579 Ki = 9.5 nM T78198 CB20NH 136144119 Ki = 5.9 nM T78198 CV4BF5 136144120 Ki = 0.25 nM T78198 C0SG1R 136144121 Ki = 0.22 nM T78198 CH5RE3 136179526 Ki = 4.7 nM T78198 CW5J3E 136179530 Ki = 415 nM T78198 CKAW94 136179532 Ki = 250 nM T78198 C1Y6QV 136179619 Ki = 1.4 nM T78198 C4O2PF 136491910 Ki = 2000 nM T78198 CY3ZK6 136491911 Ki = 2900 nM T78198 C50AHW 155569634 Ki = 180 nM T78198 D04AWP 135398631 Ki = 1500000 nM T78198 D07BNM 135460987 Ki = 10.8 nM T78198 D07VEW 135415984 Ki = 0.007 nM T78198 D0A9WP 135445969 Ki = 0.029 nM T78198 D0E6BI 135509131 Ki = 4.9 nM T78198 D0FI2L 135518164 IC50 = 1330 nM T78198 D0R5RF 135981935 Ki = 6 nM T78198 D0R6UA 135421887 IC50 = 600 nM T78198 D0SO9G 136002688 Ki = 303 nM T78198 D0T4HR 135408972 Ki = 200 nM T68334 CUR6Q3 2741928 IC50 > 16500 nM T68334 CF75UI 2837084 EC50 = 4400 nM T68334 C5HY4Z 10030777 EC50 = 2.7 nM T68334 CA5CV3 10099401 EC50 = 1.2 nM T68334 C14JLZ 10120470 EC50 = 1.7 nM T68334 CD05XM 10142987 EC50 = 3 nM T68334 CV8D5S 10164519 EC50 = 13 nM T68334 C1AZX7 10165009 EC50 = 3900 nM T68334 C1D5AE 10185204 EC50 = 400 nM T68334 C5KEB2 10461880 EC50 = 260 nM T68334 CWR47A 11156384 IC50 = 240 nM T68334 CQH9T2 11190706 IC50 = 166 nM T68334 CBX46O 11190814 IC50 = 7 nM T68334 C9U4TK 11203161 IC50 = 30 nM T68334 C0ROX1 11224637 IC50 = 31 nM T68334 CV1P0D 11224817 IC50 = 930 nM T68334 CW02AD 11258158 IC50 = 27 nM T68334 CV4JF3 11260332 IC50 = 4 nM T68334 C9NOQ3 11283209 IC50 = 9 nM T68334 CU26XM 11283470 IC50 = 5 nM T68334 C7QDK6 11306348 IC50 = 25 nM T68334 CC69SF 11352881 IC50 = 170 nM T68334 CY46FH 11373573 IC50 = 76 nM T68334 CL0X1W 11375523 IC50 = 50 nM T68334 CFTD31 11396885 IC50 = 5 nM T68334 C7AX8R 11407702 IC50 = 580 nM T68334 CKN76R 11431176 IC50 = 2800 nM T68334 C7T6IG 11442786 IC50 = 1880 nM T68334 CUGJ81 11443213 IC50 = 54 nM T68334 CRXO16 29993669 IC50 > 16500 nM T68334 CY5P9C 29993670 IC50 > 16500 nM T68334 CLVX83 44255904 EC50 = 397 nM T68334 CS29GM 44292698 EC50 = 900 nM T68334 CT5I6L 44292731 EC50 = 3.6 nM T68334 CJM9I2 44292821 EC50 > 20000 nM T68334 CJOV32 44292891 EC50 = 1600 nM T68334 C5QW1N 44292917 EC50 = 150 nM T68334 CIUV65 44292920 EC50 = 68 nM T68334 CU2A9K 44292921 EC50 > 20000 nM T68334 C7U9VP 44292938 EC50 = 14 nM T68334 C9GQD0 44292995 EC50 = 3000 nM T68334 C5EBQ8 44293018 EC50 = 3300 nM T68334 CGL93Q 44293019 EC50 = 1200 nM T68334 CDA23E 44293020 EC50 = 100 nM T68334 CH1SY2 44293169 EC50 = 1.8 nM T68334 C2C8IP 44293172 EC50 = 9.7 nM T68334 CL9RA5 44293189 EC50 = 7.2 nM T68334 C9RXK1 44293201 EC50 > 20000 nM T68334 CAHK24 44293203 EC50 = 8.9 nM T68334 CZO37J 44293287 EC50 = 120 nM T68334 CO6M1B 44293289 EC50 = 25 nM T68334 C1WC2B 44293299 EC50 = 5000 nM T68334 CUXK95 44293300 EC50 = 9000 nM T68334 C1ZSD7 44293310 EC50 > 50000 nM T68334 CV2I6P 44293324 EC50 = 2300 nM T68334 C1G9ST 44580873 EC50 = 5000 nM T68334 CK7I4M 53318154 IC50 = 39 nM T68334 C7WMT6 53320758 IC50 = 920 nM T68334 CH4JK8 53322111 EC50 = 126 nM T68334 C2Q3EJ 53324742 IC50 = 1662 nM T68334 C1Q5IF 53324743 IC50 = 1023 nM T68334 C1O7BF 53326035 IC50 = 324 nM T68334 CT8OB0 71224515 EC50 = 100 nM T68334 C3FKJ7 71224673 EC50 = 554000 nM T68334 CNK60B 71224679 EC50 = 53000 nM T68334 CVRC85 71224688 EC50 = 199000 nM T68334 C14ICS 71224861 EC50 = 8820000 nM T68334 CIOW63 71233904 EC50 < 100 nM T68334 CZN19A 71233906 EC50 = 129000 nM T68334 CS4OQ3 71233908 EC50 = 30000 nM T68334 C6TE7U 71233909 EC50 = 494000 nM T68334 CST7F4 71233912 EC50 = 508000 nM T68334 CM2A6C 71233930 EC50 = 185000 nM T68334 CUR36H 71233958 EC50 = 250000 nM T68334 C14PLX 71233981 EC50 = 100 nM T68334 CO9IW5 71234030 EC50 = 184000 nM T68334 CL8D1Q 71234037 EC50 = 28000 nM T68334 CX20JS 71234040 EC50 = 88000 nM T68334 CGA67X 71234065 EC50 = 46000 nM T68334 CFN17R 71234066 EC50 = 129000 nM T68334 CLJ5X6 71234072 EC50 = 1850000 nM T68334 CEV31L 71234099 EC50 = 184000 nM T68334 CCT2I6 71234104 EC50 = 153000 nM T68334 CWM5G4 71234119 EC50 = 1440000 nM T68334 C6ZJ9Y 71234120 EC50 = 1001000 nM T68334 CG09PV 71234266 EC50 < 100 nM T68334 C0IKJ8 71234519 EC50 < 100 nM T68334 CTDX91 71450781 EC50 = 50 nM T68334 CP5WH1 71457922 EC50 = 1 nM T68334 CO9TE5 71488103 EC50 < 100 nM T68334 C9T7SR 90656078 EC50 = 4900000 nM T68334 CG2NH6 139600336 IC50 > 16000 nM T68334 C0HN5J 139600337 IC50 > 16000 nM T87675 D05LKP 5215 IC50 = 21000 nM T87675 D07NVU 9829523 IC50 = 80 nM T87675 D07VLY 31703 IC50 = 40 nM T87675 D0E6XR 3062316 IC50 = 2633 nM T87675 D0J9ZR 4477 IC50 = 54100 nM T87675 D0R0MW 5329102 IC50 = 1837 nM T87675 D0W5HK 216239 IC50 = 3800 nM T87675 D0Y9ZE 4197 Ki > 100000 nM T87675 D00DRL 44137946 IC50 = 290 nM T87675 D00LGR 56839178 IC50 = 3 nM T87675 D02RJY 11442891 Ki = 2.5 nM T87675 D02XNW 5494449 IC50 = 0.24 nM T87675 D03HUX 49792852 IC50 > 10000 nM T87675 D03LWG 53235510 IC50 > 10000 nM T87675 D05PZB 135398495 IC50 = 3 nM T87675 D07DTV 11338033 IC50 > 10000 nM T87675 D07EHV 44814409 IC50 > 10000 nM T87675 D07HPJ 11476171 IC50 > 10000 nM T87675 D07KYT 24889392 IC50 > 10000 nM T87675 D08HOM 46207586 IC50 = 12 nM T87675 D0A5MC 11712649 IC50 = 1 nM T87675 D0CY1B 6420138 Ki = 8 nM T87675 D0E3TC 44259 IC50 < 1 nM T87675 D0EJ3B 24856041 IC50 = 5 nM T87675 D0FD6D 11751922 IC50 = 42 nM T87675 D0H2HZ 60194098 IC50 > 50118.72 nM T87675 D0IQ0Z 46885626 Ki = 490 nM T87675 D0J6AB 24748204 IC50 = 0.046 nM T87675 D0M9QZ 11485656 IC50 = 760 nM T87675 D0O0LS 25141092 IC50 = 215 nM T87675 D0P1CV 46191454 IC50 > 10000 nM T87675 D0Q7RE 16007391 Ki = 1400 nM T87675 D0Q9UX 16718576 IC50 = 1051 nM T87675 D0S4JK 24771867 IC50 = 0.04 nM T87675 D0S7HM 16041424 IC50 = 14 nM T87675 D03BNU 59604787 IC50 > 10000 nM T87675 D0A3MV 448014 IC50 > 100000000 nM T87675 D0H7AC 51346455 IC50 = 0.8 nM T87675 D0T3ME 156422 IC50 > 30000 nM T87675 C2LR7Y 1870 IC50 > 100000 nM T87675 CO2Y3R 3698 Ki = 393900 nM T87675 CW3VJ0 55970 IC50 = 79.4 nM T87675 C63WLY 89644 IC50 = 1.3 ug.mL-1 T87675 C5JE2Z 104860 IC50 = 1.7 ug.mL-1 T87675 CK8R2P 119131 Ki = 125200 nM T87675 C28CSW 158883 IC50 = 2140 nM T87675 CI1NA5 159926 IC50 = 1.9 ug.mL-1 T87675 CYBA43 177458 IC50 = 3 ug.mL-1 T87675 CQ01JA 322353 Ki = 361000 nM T87675 CQ06DW 353592 IC50 > 17000 nM T87675 CB9F1O 447961 Ki = 73 nM T87675 C6A3LY 447962 Ki = 6.9 nM T87675 C76XNU 643953 IC50 > 3000 nM T87675 CCG0B1 645436 IC50 = 300 nM T87675 CR56MT 667926 IC50 = 80 nM T87675 CQBY39 693946 IC50 = 5.559 nM T87675 C98SFI 698343 IC50 = 5.1 nM T87675 C0X8MW 779302 IC50 = 256 nM T87675 C7T1NS 802942 IC50 = 130 nM T87675 C9OYC2 802952 IC50 = 680 nM T87675 CB27WS 849733 IC50 > 10000 nM T87675 CCBR52 948954 IC50 = 423 nM T87675 CIA3X9 954308 IC50 = 200 nM T87675 CE9S3T 1164022 IC50 = 98700 nM T87675 CZ7O1H 1206526 IC50 = 2780 nM T87675 CK6Y0F 1214627 IC50 = 120 nM T87675 CX3L4O 1214628 IC50 = 25 nM T87675 CQ43JT 1214629 IC50 = 39 nM T87675 C69MXN 1214657 IC50 = 51 nM T87675 C07ZOJ 1217387 IC50 = 840 nM T87675 CHX2W6 1217619 IC50 = 1330 nM T87675 C3C7SN 1251356 IC50 = 1766 nM T87675 C92TEX 1340212 IC50 = 2650 nM T87675 CZ4W9A 1340223 IC50 = 1450 nM T87675 C8V2LG 1340269 IC50 = 12370 nM T87675 CUM36L 1340986 IC50 = 7320 nM T87675 C1N6PA 1342673 IC50 = 4790 nM T87675 CHA6M7 1343237 IC50 = 7250 nM T87675 C5GHV3 1398004 IC50 = 31300 nM T87675 C4WFP1 1587957 IC50 = 309 nM T87675 C5QD4Y 2175822 IC50 = 5710 nM T87675 CDVU98 2175921 IC50 = 5590 nM T87675 CJ4AI7 2369334 IC50 = 2100 nM T87675 C86LNP 2779952 IC50 > 100000 nM T87675 C7E4CV 2813284 IC50 = 560 nM T87675 CVW7S1 3008640 IC50 = 490 nM T87675 C4OQK8 3124004 IC50 = 5090 nM T87675 C40UDZ 3241232 IC50 = 3311 nM T87675 CB6R5K 3722581 Ki = 870 nM T87675 C43UXI 4388543 IC50 = 6600 nM T87675 C5MG8K 4663984 IC50 = 18.3 nM T87675 CEU1N6 5056270 IC50 > 100000 nM T87675 CQ8U7S 5205832 IC50 = 570 nM T87675 CI8B0V 5271602 IC50 = 34 nM T87675 CFW19M 5329009 IC50 = 6500 nM T87675 CDQ3M7 5359485 IC50 = 0.73 ug.mL-1 T87675 C54BYP 5360741 IC50 = 5 ug.mL-1 T87675 CC1VU0 5455866 IC50 = 9000 nM T87675 C1S9EH 5455880 IC50 = 390 nM T87675 C84DGA 5494424 IC50 = 0.8 nM T87675 C6P2HQ 7040530 IC50 = 3570 nM T87675 CY20RA 7458031 IC50 > 100000 nM T87675 C80NBL 7732874 IC50 = 2340 nM T87675 CM1NP6 7947603 IC50 = 420 nM T87675 CQ57EC 9548013 IC50 > 100000 nM T87675 CZCQ87 9566394 IC50 = 15140 nM T87675 C9TAL6 9826308 IC50 = 4800 nM T87675 CBGE59 9833337 IC50 = 1700 nM T87675 C23CLR 9857034 IC50 = 2310 nM T87675 C1QM0N 9858715 Ki = 17 nM T87675 C8BEZ2 9862708 IC50 = 6000 nM T87675 CUG5J1 9901007 Ki = 81 nM T87675 C7UIP5 9901505 Ki = 36 nM T87675 C2AYQ3 9924047 Ki = 86 nM T87675 CA05BZ 9925230 Ki = 9 nM T87675 CN0AJ9 9934347 IC50 = 4 nM T87675 CY0FT2 9946460 IC50 = 128 nM T87675 CDT67L 9947412 Ki = 4 nM T87675 C1BX7I 9958417 Ki = 65 nM T87675 C75QCM 9969776 Ki = 24 nM T87675 CVE1W8 10024433 Ki = 8.2 nM T87675 CRQ01L 10094689 IC50 = 1 nM T87675 CKO01Z 10094732 IC50 = 1.7 nM T87675 CZV3U5 10111694 Ki = 5 nM T87675 C06LKI 10111728 IC50 = 130 nM T87675 C3FBE4 10112131 IC50 = 5 nM T87675 CV9B4X 10112611 Ki < 1 nM T87675 CD6GN4 10113529 Ki < 1 nM T87675 CCS0B9 10128386 Ki = 690 nM T87675 CLA2N6 10133600 Ki = 6 nM T87675 CKL3V4 10134576 Ki = 1 nM T87675 C10WRQ 10153234 Ki = 55 nM T87675 CZR2G0 10156505 IC50 = 41 nM T87675 CV73FD 10157920 Ki = 2 nM T87675 CQN8M3 10159519 Ki = 2 nM T87675 CY13QK 10175096 Ki = 2 nM T87675 CR80BV 10175126 Ki = 94 nM T87675 C3QNO1 10177287 IC50 = 2120 nM T87675 CQ6J1C 10179215 Ki = 3 nM T87675 CC78NE 10179293 IC50 > 5000 nM T87675 C3KHT0 10179373 Ki = 1 nM T87675 CXD4Z2 10180161 Ki < 1 nM T87675 CO08KZ 10182284 Ki = 9 nM T87675 C8O1FV 10196735 Ki = 1 nM T87675 CFUY91 10196758 Ki = 18 nM T87675 C7PEG0 10200408 Ki = 4 nM T87675 C1Z6EJ 10222721 Ki = 2 nM T87675 C9FV7Z 10239608 Ki = 190 nM T87675 CZS9G0 10239769 Ki = 360 nM T87675 CSG14T 10239873 Ki = 39 nM T87675 C2PLB1 10239891 Ki = 87 nM T87675 C1KX3P 10248401 Ki = 4 nM T87675 CX7PD0 10252549 IC50 = 1.6 nM T87675 CGF6I3 10267834 Ki = 24 nM T87675 C28AEC 10268530 Ki = 20 nM T87675 CLQ3P2 10270356 Ki = 5 nM T87675 C13VMD 10273410 Ki = 2.4 nM T87675 CJGH26 10275985 IC50 > 5000 nM T87675 C9V3SL 10289802 Ki = 220 nM T87675 CF9N7Y 10292186 Ki = 24 nM T87675 CNT46L 10311867 Ki = 110 nM T87675 CA23IN 10311891 Ki = 220 nM T87675 CD63MH 10312249 Ki = 280 nM T87675 C9J3RM 10320107 Ki = 12 nM T87675 CB45DL 10322308 IC50 < 1 nM T87675 CMY9D2 10340715 Ki = 14 nM T87675 CG2L4Z 10343860 IC50 = 1.6 nM T87675 CJ5W7O 10388447 IC50 = 3.7 nM T87675 CHLW70 10412796 IC50 < 1 nM T87675 C7HBP6 10429593 IC50 > 10000 nM T87675 CC3L8Z 10430000 Ki = 19 nM T87675 C41GHN 10435854 IC50 = 1.3 nM T87675 CASV91 10466228 IC50 = 29000 nM T87675 C1H7OM 11167062 IC50 = 100 nM T87675 C8T2NG 11211389 IC50 = 6800 nM T87675 CQ4XT3 11224593 IC50 = 8300 nM T87675 CK6U2S 11249084 IC50 = 27 nM T87675 CJL85B 11261882 IC50 > 50000 nM T87675 CBOP58 11293798 Ki > 10000 nM T87675 C3F6UB 11300082 IC50 > 10000 nM T87675 C95HYJ 11305344 IC50 = 130 nM T87675 CT5NM2 11353953 IC50 = 94 nM T87675 CE8VP2 11361885 IC50 = 4200 nM T87675 C26BZX 11362471 Ki > 10000 nM T87675 CB45PJ 11362483 IC50 = 7200 nM T87675 C4IH5E 11383525 IC50 = 8300 nM T87675 CKLC82 11384622 IC50 = 160 nM T87675 CWXB93 11397177 Ki > 10000 nM T87675 CT3VP7 11398307 IC50 = 764 nM T87675 CWM18I 11406175 IC50 > 10000 nM T87675 CFOZ52 11407074 IC50 > 10000 nM T87675 C25NHJ 11416146 IC50 > 10000 nM T87675 C1WXC5 11417488 IC50 = 3229 nM T87675 CFJ6B2 11441375 IC50 = 2000 nM T87675 CLZ3M8 11442557 IC50 = 6 nM T87675 CM21YJ 11453049 IC50 = 1258.93 nM T87675 C4Q7XD 11474276 IC50 = 5000 nM T87675 C9LA1E 11486283 IC50 > 10000 nM T87675 C2Z7WP 11486459 IC50 = 1500 nM T87675 C74BAE 11487958 IC50 = 24 nM T87675 C1UFM0 11497983 Ki = 1368 nM T87675 CBW4Q3 11500669 IC50 = 1000 nM T87675 CCVX84 11501979 IC50 = 67 nM T87675 C5NQ0Y 11502548 IC50 = 43 nM T87675 C4VFT0 11504974 IC50 < 1 nM T87675 CRS73J 11505438 IC50 = 12 nM T87675 CR7MJ1 11508531 IC50 = 14 nM T87675 CTF2B7 11512480 IC50 < 1 nM T87675 CV1YT6 11519624 IC50 < 0.1 nM T87675 CMP85Z 11519853 IC50 = 106 nM T87675 CU4J8R 11523891 IC50 = 28 nM T87675 CCU8G9 11526006 IC50 = 18 nM T87675 C1WV7U 11527003 IC50 < 1 nM T87675 CL7X4Q 11530963 IC50 = 5400 nM T87675 C3KNI0 11533732 IC50 > 1000 nM T87675 CAWT72 11537541 IC50 = 29 nM T87675 CTG83F 11539329 Ki > 6900 nM T87675 C6ZY9F 11545541 IC50 = 93 nM T87675 C0WXA4 11548214 IC50 = 5 nM T87675 CZ3D4J 11548500 IC50 < 1 nM T87675 C26ABY 11551547 IC50 = 66 nM T87675 CZL4V1 11558640 IC50 = 2500 nM T87675 CACS26 11561968 Ki > 1000 nM T87675 CH05WP 11566279 IC50 = 640 nM T87675 C26ZYU 11577723 IC50 < 1 nM T87675 CHR4Q6 11580435 IC50 = 570 nM T87675 CO9KP5 11583459 IC50 > 10000 nM T87675 C2CT6L 11587983 IC50 = 65 nM T87675 C8E5DA 11589674 IC50 = 931 nM T87675 CMIL86 11590363 Ki > 6900 nM T87675 C5QF4P 11592171 IC50 = 55 nM T87675 COV9L6 11598217 IC50 = 1 nM T87675 CKJ52I 11599631 IC50 = 452 nM T87675 CJ42AE 11603072 IC50 = 49 nM T87675 C9WG0V 11604623 IC50 = 600 nM T87675 C5ER3Q 11611230 IC50 = 56 nM T87675 CF34LT 11613706 IC50 = 578 nM T87675 C5U4XY 11617275 IC50 = 93 nM T87675 CUVW54 11617466 IC50 = 36 nM T87675 CQBU93 11620791 IC50 = 472 nM T87675 C4U7HM 11621097 IC50 = 15 nM T87675 CI8CR3 11623444 Ki = 3300 nM T87675 CG6UC2 11624169 IC50 = 37 nM T87675 C7JDC2 11628500 IC50 = 2 nM T87675 CZ25EP 11631251 Ki > 100000 nM T87675 CIWA03 11632150 Ki = 0.4 nM T87675 CAN9R0 11632327 IC50 = 1600 nM T87675 C5Z1YR 11633940 IC50 = 6 nM T87675 CL53BK 11639104 IC50 = 32 nM T87675 C9T6SC 11640926 Ki > 6900 nM T87675 COF4I7 11645638 IC50 = 24 nM T87675 CEV5X2 11646645 Ki = 5 nM T87675 C6LK9N 11646783 Ki = 14900 nM T87675 C2CVI7 11647020 Ki = 3 nM T87675 CEBS68 11652621 IC50 = 31 nM T87675 CKR96C 11653244 IC50 = 120 nM T87675 C85HAQ 11655501 IC50 = 170 nM T87675 CPNM76 11658909 IC50 = 270 nM T87675 CX89MN 11663832 IC50 = 1 nM T87675 C0PM2W 11664170 IC50 < 1 nM T87675 C8XGK5 11667761 IC50 = 25 nM T87675 C8TO6F 11668744 IC50 = 420 nM T87675 C8Z1YO 11681497 IC50 = 23 nM T87675 CPQ19H 11681507 IC50 = 270 nM T87675 CJ9KN7 11683817 IC50 > 10000 nM T87675 CKC51F 11689306 IC50 = 550 nM T87675 CU0E8O 11690457 Ki > 10000 nM T87675 CTG83S 11692745 IC50 < 1 nM T87675 CIN01S 11692746 IC50 = 111 nM T87675 C5SBN0 11699912 IC50 = 483 nM T87675 C5R4NP 11705035 IC50 = 0.9 nM T87675 CB0AP2 11705863 Ki > 1000 nM T87675 CFX9V2 11709165 IC50 = 115 nM T87675 CH7DO8 11710518 IC50 = 240 nM T87675 C0YF7W 11713454 IC50 = 158 nM T87675 C8P3BC 11716968 IC50 = 17 nM T87675 CW1VX7 11717761 IC50 = 109 nM T87675 C93KHF 11718021 Ki = 1 nM T87675 CJSV21 11744184 Ki = 9.2 nM T87675 CS5QL4 11749561 IC50 = 3600 nM T87675 CV64JS 11750694 IC50 = 4400 nM T87675 CVFS29 11751305 IC50 = 65 nM T87675 C5S6LY 11846197 IC50 = 32 nM T87675 CG5VI7 11846198 IC50 = 59 nM T87675 C6Y1BN 11846199 IC50 = 48 nM T87675 CB89CN 11846366 IC50 = 13 nM T87675 C6B7WH 11846367 IC50 = 10 nM T87675 CU6YB5 11846701 IC50 = 6 nM T87675 CTH1S7 11846702 IC50 = 66 nM T87675 CMG3D0 11846703 IC50 = 48 nM T87675 COQ1V5 11846875 IC50 = 52 nM T87675 CQ8A5O 11846876 IC50 = 45 nM T87675 CJ3Y5L 11846877 IC50 = 31 nM T87675 CI8Q5T 11846878 IC50 = 9 nM T87675 C7VN3I 11847026 IC50 = 11 nM T87675 CD6BP5 11847027 IC50 = 5 nM T87675 CNW69R 11847028 IC50 = 83 nM T87675 C73VNF 11847342 IC50 = 25 nM T87675 C9JT4S 11847343 IC50 = 18 nM T87675 C3VFC0 11847344 IC50 = 27 nM T87675 CHR92S 11858109 IC50 > 200 nM T87675 CT0H7I 11949628 Ki = 2 nM T87675 CUDO23 11994441 IC50 = 354 nM T87675 C6H2RT 11994444 IC50 = 9 nM T87675 CN4JP1 11994445 IC50 = 452 nM T87675 CM50UH 12000646 IC50 = 82 nM T87675 CGJ69E 12000661 IC50 = 17 nM T87675 C7Y8MZ 12342815 IC50 = 5540 nM T87675 CKJ12Y 12650481 IC50 = 12500 nM T87675 CJD06E 12773351 IC50 = 6500 nM T87675 C86IBL 12799331 Ki > 100000 nM T87675 CP4C7R 12799333 Ki > 100000 nM T87675 C0QGS1 13942472 Ki = 184700 nM T87675 CY30ZN 14293776 IC50 = 3000 nM T87675 CDGF78 15282555 IC50 = 100 nM T87675 C7LB4I 15949613 IC50 = 1050 nM T87675 CFPW41 16007116 Ki > 6900 nM T87675 CQR5O7 16042971 IC50 = 350 nM T87675 C9TU1O 16046126 IC50 > 1000 nM T87675 CW18IV 16070056 IC50 = 640 nM T87675 CKR57M 16086104 IC50 > 5000 nM T87675 C16NRY 16086114 IC50 > 5000 nM T87675 CQG45C 16109001 IC50 = 25000 nM T87675 C5VPH9 16129448 IC50 = 472 nM T87675 C8FLH6 16202152 IC50 = 42 nM T87675 CG5PZ4 16221284 Ki = 18 nM T87675 CUQ5O3 16221285 Ki = 14 nM T87675 C2XK5Y 16221286 Ki = 30 nM T87675 CL3VC4 16221338 Ki = 83 nM T87675 CF7YG2 16221339 Ki = 140 nM T87675 C6Q7FT 16221340 Ki = 13 nM T87675 C1BVO9 16221341 Ki = 160 nM T87675 CLX80H 16221342 Ki = 350 nM T87675 CIA5Y4 16221343 Ki = 950 nM T87675 CG9W2O 16221393 Ki = 980 nM T87675 CYJZ19 16221394 Ki = 1400 nM T87675 CRV7C8 16221627 Ki = 2 nM T87675 C4FUV3 16221628 Ki = 8 nM T87675 C6GHV5 16221629 Ki = 39 nM T87675 CB57GO 16221630 Ki = 9 nM T87675 CCT7I4 16666303 IC50 > 10000 nM T87675 CAK1C4 16666757 IC50 > 100000 nM T87675 C1QRG8 16666806 IC50 = 21230 nM T87675 CF8B5S 16666857 IC50 = 338 nM T87675 C5U8LG 16666858 IC50 = 205 nM T87675 CJ9C7N 16666859 IC50 = 200 nM T87675 C5JQ6H 16666860 IC50 = 179 nM T87675 C4VW0O 16666861 IC50 = 135 nM T87675 C1IO4K 16666862 IC50 = 100 nM T87675 CS1LR2 16666908 IC50 = 100 nM T87675 CI32LX 16666909 IC50 = 90 nM T87675 C07BIL 16666910 IC50 = 338 nM T87675 C71TSX 16666911 IC50 = 44 nM T87675 CKT4N2 16719269 Ki = 2.4 nM T87675 CY1E2N 16723801 IC50 > 100000 nM T87675 CDVO81 16730408 IC50 = 13 nM T87675 CQ5H0C 16730410 IC50 = 79 nM T87675 C5D2NG 16730500 IC50 = 240 nM T87675 CPUN56 16730501 IC50 = 200 nM T87675 C38ZAH 16730583 IC50 > 10000 nM T87675 CU5W8H 16730586 IC50 = 1900 nM T87675 CTX68K 16730664 IC50 = 91 nM T87675 CMFL15 16730666 IC50 = 620 nM T87675 C23VWJ 16731303 IC50 = 140 nM T87675 C6S3YO 16731782 IC50 = 16 nM T87675 CK9CV4 16733534 IC50 = 28 nM T87675 C5M1EL 20399253 Ki = 21300 nM T87675 C5NCJ3 20604194 Ki = 5.1 nM T87675 CL81VC 21100709 IC50 = 1340 nM T87675 C0KH4J 21106464 IC50 = 100 nM T87675 CI4GS3 21106477 IC50 = 35 nM T87675 CBL7W3 21106491 IC50 = 720 nM T87675 C5W9CM 21106492 IC50 = 71 nM T87675 CF59EQ 21106541 IC50 = 650 nM T87675 C1HXU3 21506922 IC50 = 4300 nM T87675 C1N4XZ 21874004 IC50 = 13 nM T87675 C8IF5U 21991073 Ki = 17 nM T87675 CD45BA 22060262 IC50 = 30 nM T87675 CL37GA 22426194 IC50 > 100000 nM T87675 C3XI0R 23339828 Ki = 99500 nM T87675 C4V9UD 23545854 Ki = 10 nM T87675 CP01RM 23583059 IC50 = 35 nM T87675 C29OFZ 23585419 IC50 = 365 nM T87675 C0VQ4E 23585422 IC50 = 55 nM T87675 C63DWY 23585534 IC50 = 81 nM T87675 CQ53UI 23585535 IC50 = 81 nM T87675 CXH58R 23586142 IC50 = 3110 nM T87675 C3YK5H 23644668 IC50 = 3900 nM T87675 CV9I6B 23645979 IC50 = 2140 nM T87675 C8N0IA 23645980 IC50 > 10000 nM T87675 C0J6OK 23645981 IC50 = 660 nM T87675 C7SP6F 23645982 IC50 = 8500 nM T87675 CNP20Z 23645983 IC50 = 4850 nM T87675 C4TW1K 23645984 IC50 > 10000 nM T87675 C5SPY4 23645985 IC50 = 440 nM T87675 CO0DL7 23645986 IC50 = 160 nM T87675 C2A9UN 23645987 IC50 = 390 nM T87675 CJVQ86 23645988 IC50 > 10000 nM T87675 C7IRF0 23645989 IC50 > 10000 nM T87675 CQIU74 23645990 IC50 > 10000 nM T87675 CLD4U6 23645991 IC50 > 10000 nM T87675 CTR39K 23645992 IC50 > 10000 nM T87675 CHM34D 23646072 IC50 = 3 nM T87675 C2KW3S 23646073 IC50 = 629 nM T87675 CV5M8N 23646074 IC50 = 0.15 nM T87675 CH58XV 23646075 IC50 = 70 nM T87675 C3W8UV 23646076 IC50 = 85 nM T87675 C0J8GT 23646077 IC50 = 690 nM T87675 C35CBJ 23646078 IC50 = 17 nM T87675 CQHK69 23646624 IC50 = 47 nM T87675 CH1B7R 23646625 IC50 = 49 nM T87675 CF9CH8 23646627 IC50 = 0.6 nM T87675 C8TIN5 23646628 IC50 = 12 nM T87675 C9ZS1H 23646629 IC50 = 39 nM T87675 C50QUN 23646630 IC50 = 18 nM T87675 CS3UY4 23646631 IC50 = 13 nM T87675 CR7JY4 23646632 IC50 = 9 nM T87675 CIM15C 23646633 IC50 = 18 nM T87675 C1TZ4I 23647263 IC50 = 57.6 nM T87675 CS69KN 23647269 IC50 = 11.3 nM T87675 CS9CG0 23729140 IC50 = 3.8 nM T87675 CNO0H1 23909187 IC50 = 1620 nM T87675 CFMQ08 24370907 IC50 > 100000 nM T87675 CHU49V 24757938 IC50 = 371 nM T87675 CQNP54 24764449 IC50 = 1000 nM T87675 CCPS81 24764502 IC50 > 35000 nM T87675 C8LA5E 24767906 IC50 = 1.2 nM T87675 CY3ZM6 24767908 IC50 = 3.7 nM T87675 C3ZRQ5 24767909 IC50 = 2.1 nM T87675 CGU7L3 24767910 IC50 = 6.3 nM T87675 C04EBZ 24767923 IC50 = 0.27 nM T87675 CMQ9N4 24767924 IC50 = 5.1 nM T87675 C4Z9CN 24769780 IC50 = 426 nM T87675 CXSZ08 24783396 Ki = 0.59 nM T87675 C74EZB 24815963 IC50 = 53 nM T87675 CEC8T9 24815964 IC50 = 128 nM T87675 C2EC0A 24815965 IC50 = 495 nM T87675 CIWJ29 24815966 IC50 = 514 nM T87675 C75MAH 24816055 IC50 = 39 nM T87675 CIC7O1 24816056 IC50 = 414 nM T87675 CO9Z0H 24822598 IC50 = 840 nM T87675 C51IZL 24822599 IC50 = 620 nM T87675 CA90EF 24822600 IC50 = 3600 nM T87675 C4A6LB 24823090 IC50 = 560 nM T87675 C2B4JP 24823091 IC50 = 3700 nM T87675 CF6M3W 24823093 IC50 = 8300 nM T87675 C0NLO8 24823094 IC50 = 8300 nM T87675 C7D8PC 24823095 IC50 = 8300 nM T87675 C14FLQ 24823250 IC50 = 930 nM T87675 C3KPO7 24823251 IC50 = 3500 nM T87675 C36BFD 24823252 IC50 = 25000 nM T87675 CBF60S 24823253 IC50 = 8300 nM T87675 C84VZK 24824448 IC50 = 440 nM T87675 C6OC4K 24824449 IC50 = 1700 nM T87675 C3RCV4 24855973 IC50 = 60 nM T87675 C3GP7H 24880024 IC50 = 22 nM T87675 C2AB7C 24893974 IC50 = 2900 nM T87675 C4V9GH 24894117 IC50 = 16000 nM T87675 CJH19T 24894883 IC50 = 3200 nM T87675 CJ14YB 24894884 IC50 = 16000 nM T87675 C57BHF 24894888 IC50 = 29000 nM T87675 CB5TP8 24894992 IC50 = 30000 nM T87675 CP7QT2 24894995 IC50 = 3200 nM T87675 C41SIT 24894996 IC50 = 33000 nM T87675 CFW40U 24894997 IC50 = 6500 nM T87675 CF4N9X 24895100 IC50 = 47000 nM T87675 CY8L7E 24896769 IC50 > 10000 nM T87675 CN13JF 24899915 IC50 = 0.39 ug.mL-1 T87675 CBWR97 24899916 IC50 = 1.5 ug.mL-1 T87675 C9F2JD 24899917 IC50 > 10 ug.mL-1 T87675 C64MTI 24900160 IC50 = 2.7 ug.mL-1 T87675 CO2I6Q 24900161 IC50 = 4.4 ug.mL-1 T87675 CT8OF0 24983254 IC50 = 141 nM T87675 CVF62Q 24983255 IC50 = 380 nM T87675 CX6FR3 24983298 IC50 = 1067 nM T87675 CEQ1F2 24983299 IC50 = 327 nM T87675 CQ46VT 24983495 IC50 = 19 nM T87675 CQEV29 24992861 IC50 = 605 nM T87675 CCZF80 24992862 IC50 = 2900 nM T87675 CU5B6R 24992864 IC50 > 10000 nM T87675 C4EG8R 24993189 IC50 > 10000 nM T87675 C3DI7Y 24995523 IC50 = 9 nM T87675 CJ5GM7 25008277 IC50 = 5600 nM T87675 CHLQ49 25063262 IC50 > 100000 nM T87675 C2KY1G 25094210 IC50 <= 4 nM T87675 CR7X4M 25094243 IC50 = 22 nM T87675 CA6E0J 25094245 IC50 = 105 nM T87675 CC5NE0 25094283 IC50 = 85 nM T87675 CTV54O 25123227 IC50 = 2900 nM T87675 CG3XC9 25124150 IC50 = 1600 nM T87675 CO2IR5 25124816 IC50 > 1500 nM T87675 C1IYN7 25127854 IC50 = 170 nM T87675 CKD14B 25127856 IC50 = 120 nM T87675 CJBX60 25128180 IC50 > 1000 nM T87675 CC5SD9 25128181 IC50 = 680 nM T87675 CXF6T2 25138097 IC50 = 3200 nM T87675 C16OVX 25138098 IC50 > 20000 nM T87675 CKS85T 25138099 IC50 = 1200 nM T87675 CIG93H 25138100 IC50 > 20000 nM T87675 CUO0D6 25138101 IC50 = 1200 nM T87675 C0X1RB 25138102 IC50 = 250 nM T87675 C63CUY 25138103 IC50 > 20000 nM T87675 COT2Y8 25138104 IC50 = 2500 nM T87675 CH7EJ6 25138105 IC50 > 10000 nM T87675 CVKD89 25138106 IC50 = 4900 nM T87675 CWY2Q8 25138107 IC50 = 52 nM T87675 CESX32 25138108 IC50 = 7200 nM T87675 C8C2GV 25138109 IC50 = 9 nM T87675 C8QB2K 25138110 IC50 = 50 nM T87675 CXJ2W1 25138111 IC50 = 41 nM T87675 C3KLX9 25138112 IC50 = 23 nM T87675 COM5W2 25138113 IC50 = 39 nM T87675 CJ5K3Z 25138114 IC50 = 280 nM T87675 CX0RG8 25138115 IC50 = 96 nM T87675 C96IEQ 25138116 IC50 = 11 nM T87675 C8XW3Z 25138117 IC50 = 30 nM T87675 CZ07IH 25138118 IC50 = 270 nM T87675 C02EZG 25138119 IC50 = 4 nM T87675 C7LS2A 25138120 IC50 = 53 nM T87675 C80HOQ 25138349 IC50 = 3180 nM T87675 CP6G0C 25143601 IC50 < 4 nM T87675 CGT1W6 25144294 IC50 <= 4 nM T87675 C0CD4W 25144582 IC50 <= 4 nM T87675 CU7VR0 25144732 IC50 <= 4 nM T87675 CX5H1V 25145005 IC50 <= 4 nM T87675 CAO7K5 25145142 IC50 <= 4 nM T87675 CP3N2V 25145143 IC50 <= 4 nM T87675 C65YQG 25145144 IC50 <= 4 nM T87675 C6BWZ8 25145145 IC50 <= 4 nM T87675 C1VE8B 25145146 IC50 <= 4 nM T87675 CE31OI 25145147 IC50 <= 4 nM T87675 CORN76 25145280 IC50 <= 4 nM T87675 CF97LX 25145281 IC50 <= 4 nM T87675 CJ0ST3 25145282 IC50 <= 4 nM T87675 CFG67C 25145424 IC50 < 4 nM T87675 C52NQJ 25145568 IC50 < 4 nM T87675 C9N8UY 25145713 IC50 < 4 nM T87675 CX8LG5 25145714 IC50 < 4 nM T87675 C85ZKA 25145715 IC50 < 4 nM T87675 C78YWA 25145716 IC50 < 4 nM T87675 CL47VI 25145718 IC50 <= 4 nM T87675 C1PL5W 25151216 IC50 = 53 nM T87675 CO90BX 25151778 IC50 = 55 nM T87675 C9UN0X 25153410 IC50 = 10 nM T87675 C16MQN 25153621 IC50 = 30 nM T87675 CSB49J 25153624 IC50 = 10 nM T87675 C02XQS 25153836 IC50 = 10 nM T87675 C2G5TB 25153837 IC50 = 14 nM T87675 CH3M5P 25154041 IC50 = 15 nM T87675 CIUJ83 25167109 IC50 = 265 nM T87675 C0OW7X 25167905 IC50 = 156 nM T87675 CN0I2H 25174496 IC50 = 1623 nM T87675 COM37V 25174498 IC50 = 166 nM T87675 CQRJ38 25175157 IC50 = 12500 nM T87675 CU4Z9Y 25175322 IC50 > 12500 nM T87675 CCD92Y 25175326 IC50 = 12500 nM T87675 CFX81M 25175327 IC50 > 12500 nM T87675 CAN9J0 25175480 IC50 = 3790 nM T87675 CJ76ZI 25175481 IC50 = 12500 nM T87675 C2K3DU 25175482 IC50 = 586 nM T87675 C7TP4W 25175646 IC50 = 4780 nM T87675 C7K9VO 25175648 IC50 = 12200 nM T87675 CDK84B 25175951 IC50 > 12500 nM T87675 CN9B1A 25176267 IC50 = 12500 nM T87675 C5EQD8 25176269 IC50 = 12500 nM T87675 CHMK36 25176588 IC50 > 12500 nM T87675 CIB0V7 25176589 IC50 > 12500 nM T87675 CCM43R 25181368 Ki = 66900 nM T87675 C76WYH 25184035 IC50 > 10000 nM T87675 CNG96H 25210579 IC50 > 10000 nM T87675 CMRJ98 25223775 IC50 = 13740 nM T87675 CP7SL8 25223778 IC50 = 1580 nM T87675 C09RHG 25223779 IC50 = 1350 nM T87675 CC6T8S 25223869 IC50 = 804 nM T87675 CEV8A3 25223870 IC50 > 50000 nM T87675 C6ISC7 25223871 IC50 = 1484 nM T87675 C73IUG 25223872 IC50 = 1937 nM T87675 CVG73U 25223873 IC50 = 1623 nM T87675 CXT7B2 25223874 IC50 = 838 nM T87675 C3BM5I 25223875 IC50 = 1580 nM T87675 COHJ58 25223973 IC50 = 2895 nM T87675 CXQJ27 25223974 IC50 = 449 nM T87675 CY1A2C 25223975 IC50 = 1087 nM T87675 CGUS12 25223976 IC50 = 1568 nM T87675 CHG7U0 25223977 IC50 = 1447 nM T87675 CQS0E9 25223978 IC50 = 33 nM T87675 C91IOK 25224078 IC50 = 11505 nM T87675 CH95DI 25224079 IC50 = 5250 nM T87675 CTZP96 25224080 IC50 = 1942 nM T87675 CUGL97 25224081 IC50 > 50000 nM T87675 CF54MI 25224082 IC50 = 1071 nM T87675 CL4OG1 25224083 IC50 = 1746 nM T87675 C1BHN8 25224190 IC50 = 460 nM T87675 C1B7OZ 25224191 IC50 = 960 nM T87675 C2H5TW 25224192 IC50 = 719 nM T87675 CWP29U 25242324 IC50 > 10000 nM T87675 CLB28U 25271180 IC50 > 100000 nM T87675 CGHR32 25271181 IC50 > 100000 nM T87675 C3E9XU 25271513 IC50 > 100000 nM T87675 CGBX14 25271514 IC50 = 100000 nM T87675 C76NWM 25271515 IC50 > 100000 nM T87675 C6C4YR 25271516 IC50 > 100000 nM T87675 CUAK50 25271517 IC50 > 100000 nM T87675 CIR67H 25271518 IC50 > 10000 nM T87675 COX1N3 27460865 IC50 > 100000 nM T87675 C2U0NP 30291209 IC50 > 100000 nM T87675 C7S6OT 30291292 IC50 > 100000 nM T87675 CRH7O2 42628076 IC50 = 6 nM T87675 CM5QJ4 42628077 IC50 = 4.3 nM T87675 CJ5U1X 42639664 IC50 = 2.8 ug.mL-1 T87675 CJHE74 42640796 Ki = 20 nM T87675 C2CTI1 44129603 IC50 = 16 nM T87675 C1IYU0 44139710 IC50 = 3.4 nM T87675 C04IJO 44139711 IC50 = 10 nM T87675 CN2G3C 44139712 IC50 = 54 nM T87675 CTN41Y 44156909 IC50 = 4400 nM T87675 CN0X1C 44156917 IC50 > 10000 nM T87675 C6CHK8 44177628 IC50 = 1828 nM T87675 CD30LF 44177630 IC50 = 836 nM T87675 CCOE96 44177727 IC50 = 434 nM T87675 CT3G5K 44177728 IC50 = 2447 nM T87675 CGV40N 44177837 IC50 = 413 nM T87675 CTVZ96 44177838 IC50 > 3000 nM T87675 C67ODN 44177840 IC50 = 57 nM T87675 CJE8L0 44177955 IC50 = 1931 nM T87675 C7JY2E 44177956 IC50 = 859 nM T87675 CU08TA 44178067 IC50 = 185 nM T87675 CO1IM5 44178068 IC50 = 186 nM T87675 CO6HU7 44178069 IC50 = 12 nM T87675 CX4R1O 44178070 IC50 = 44 nM T87675 CN8WB9 44189332 IC50 = 4 nM T87675 CK6I4N 44205288 IC50 = 7 nM T87675 CVH39F 44206601 IC50 = 70 nM T87675 CWM59J 44207068 IC50 = 4 nM T87675 CG1HI8 44207069 IC50 = 4 nM T87675 C6ZOR8 44207311 IC50 = 9 nM T87675 COAT76 44207312 IC50 = 7 nM T87675 CX1JE3 44207314 IC50 = 5 nM T87675 CAX3V9 44207547 IC50 = 2 nM T87675 CNA6M5 44207549 IC50 = 3 nM T87675 CEO05J 44207551 IC50 = 9 nM T87675 COBC24 44207552 IC50 = 9 nM T87675 C1Q6YG 44208454 IC50 = 2 nM T87675 C8KNA3 44219632 Ki = 800 nM T87675 CAF92O 44224067 IC50 = 180 nM T87675 CI46ND 44224068 IC50 = 28 nM T87675 C9T6BO 44224069 IC50 = 19 nM T87675 CLC03S 44224070 IC50 = 13 nM T87675 C7BXD4 44224071 IC50 = 9 nM T87675 CHS9Q2 44224072 IC50 = 59 nM T87675 C79UTZ 44224073 IC50 = 25 nM T87675 CP7O2F 44224074 IC50 = 140 nM T87675 CV3Q2A 44224075 IC50 = 64 nM T87675 C64ORM 44224076 IC50 = 18 nM T87675 C02FQP 44224077 IC50 = 14 nM T87675 C6W5EU 44224078 IC50 > 17000 nM T87675 C0U4DE 44224079 IC50 > 17000 nM T87675 CS5J8E 44224080 IC50 = 8 nM T87675 CTZ58V 44224081 IC50 = 14 nM T87675 CFM7U5 44224082 IC50 = 23 nM T87675 CIQ47W 44224083 IC50 = 150 nM T87675 C6SA7N 44224084 IC50 = 20 nM T87675 CNQY69 44224085 IC50 = 260 nM T87675 C1BGY0 44224086 IC50 = 78 nM T87675 C6MNV0 44224087 IC50 = 67 nM T87675 CX4J1Z 44224088 IC50 = 180 nM T87675 C2QBT5 44224089 IC50 = 75 nM T87675 C42KXR 44224090 IC50 = 160 nM T87675 C9V1KW 44224091 IC50 = 640 nM T87675 C7RDQ9 44224092 IC50 = 49 nM T87675 CC87BK 44224093 IC50 = 51 nM T87675 CSL23Q 44224094 IC50 = 19 nM T87675 C36FHU 44224095 IC50 = 78 nM T87675 CZH14J 44224096 IC50 = 36 nM T87675 CKEJ58 44224097 IC50 = 14 nM T87675 C4LNW7 44224098 IC50 = 20 nM T87675 CLJ3S6 44224099 IC50 = 50 nM T87675 C6G2EC 44232693 IC50 = 374 nM T87675 CFVC13 44232694 IC50 = 175 nM T87675 CV0FL9 44232695 IC50 = 51 nM T87675 CN0UM6 44232696 IC50 = 649 nM T87675 C4KUD5 44232697 IC50 = 1343 nM T87675 CA05LE 44232698 IC50 = 1615 nM T87675 CYCX40 44232939 IC50 = 638 nM T87675 CT1CU7 44232940 IC50 = 1437 nM T87675 C4NW9L 44232941 IC50 = 2940 nM T87675 CGTI98 44232942 IC50 > 10000 nM T87675 CCG09Z 44235884 IC50 > 10000 nM T87675 CY8A7D 44235885 IC50 = 53 nM T87675 CE42KQ 44235886 IC50 = 30 nM T87675 C5R4QP 44235887 IC50 > 10000 nM T87675 CLB67D 44235888 IC50 = 582 nM T87675 C2GRK8 44236107 IC50 = 1000 nM T87675 C4AJ7M 44236108 IC50 = 625 nM T87675 CR27YG 44236109 IC50 = 1584 nM T87675 CBN34C 44236110 IC50 = 1184 nM T87675 CS8XM3 44236111 IC50 = 535 nM T87675 CZIT93 44236112 IC50 = 855 nM T87675 C09YHS 44236349 IC50 > 5000 nM T87675 C13QXB 44236351 IC50 = 50 nM T87675 CJ37DI 44236353 IC50 = 312 nM T87675 CK5CF7 44236354 IC50 = 364 nM T87675 CYE36B 44241613 IC50 > 40000 nM T87675 C6LG5T 44241614 IC50 > 40000 nM T87675 C1I9PA 44250391 IC50 = 73.4 nM T87675 CF6SL7 44256410 IC50 = 90 nM T87675 CK78QV 44400234 IC50 = 65 nM T87675 C45LMI 44400295 IC50 = 5 nM T87675 C23EUL 44405803 IC50 > 10000 nM T87675 CPC7U9 44405842 IC50 = 3500 nM T87675 CTS08A 44405843 IC50 = 1100 nM T87675 CR0DT5 44405844 IC50 = 320 nM T87675 C9IL3J 44405863 IC50 = 1100 nM T87675 CCN1E4 44405864 IC50 = 330 nM T87675 CD3WX8 44405869 IC50 = 1900 nM T87675 CCX8K0 44405872 IC50 = 970 nM T87675 CI48BX 44405878 IC50 = 2200 nM T87675 CP3NQ2 44405895 IC50 = 470 nM T87675 CQ7WF2 44405896 IC50 = 5000 nM T87675 CVAG19 44405901 IC50 = 3700 nM T87675 C4C9SI 44405906 IC50 = 1200 nM T87675 CD92OT 44408804 IC50 = 0.8 nM T87675 C1VT7R 44417767 IC50 = 260 nM T87675 C27FEU 44417816 IC50 = 70 nM T87675 C2B4JR 44417817 IC50 = 3900 nM T87675 C9UC3V 44417819 IC50 = 6 nM T87675 C47YDK 44417820 IC50 = 0.6 nM T87675 C6DQ1Y 44433666 IC50 = 76000 nM T87675 C6RUI9 44433668 IC50 = 98000 nM T87675 C02WQZ 44433669 IC50 = 16500 nM T87675 C4E5GO 44433670 IC50 = 5900 nM T87675 CH5RU0 44433672 IC50 = 40000 nM T87675 CZC36W 44433673 IC50 = 35000 nM T87675 CY69UF 44433675 IC50 = 25000 nM T87675 CVGU29 44433676 IC50 = 9600 nM T87675 CK40JQ 44433678 IC50 = 10000 nM T87675 C52CZM 44433680 IC50 = 16000 nM T87675 CIA24G 44433681 IC50 = 4600 nM T87675 C65RIX 44433682 IC50 = 4400 nM T87675 CBKL97 44433683 IC50 = 490 nM T87675 CY5PS6 44433684 IC50 = 740 nM T87675 CSJ0N7 44433685 IC50 = 6900 nM T87675 C7BC9Q 44433686 IC50 = 20000 nM T87675 C5JSQ2 44433688 IC50 = 18000 nM T87675 C0XC7N 44433689 IC50 = 9000 nM T87675 CR2E5M 44433692 IC50 = 250 nM T87675 C5NAJ8 44433693 IC50 = 7000 nM T87675 C4B6FY 44433694 IC50 = 2400 nM T87675 C58OFB 44433695 IC50 = 870 nM T87675 CBF9P2 44447867 Ki = 340 nM T87675 CZ6G7A 44447868 Ki = 540 nM T87675 CE2D1C 44447869 Ki = 1300 nM T87675 C18TSU 44447870 Ki = 1100 nM T87675 CUH86T 44447871 Ki = 3000 nM T87675 CS2G7K 44448292 IC50 = 128 nM T87675 C4E5DN 44448294 IC50 = 112 nM T87675 CU06RO 44448295 IC50 = 85 nM T87675 CD3N2S 44448318 IC50 = 375 nM T87675 C4C2EM 44448320 IC50 = 292 nM T87675 CK6WJ8 44448397 IC50 = 346 nM T87675 C08EFA 44448716 IC50 = 910 nM T87675 C79YQL 44448738 IC50 = 7300 nM T87675 CTN76R 44450679 IC50 = 11 nM T87675 C8SLI9 44454852 IC50 = 18300 nM T87675 CJLU30 44454890 IC50 = 15200 nM T87675 CJME58 44454924 IC50 = 8000 nM T87675 C9MV2P 44468256 IC50 = 24 nM T87675 CH74FU 44470172 IC50 = 43 nM T87675 CRST03 44470317 IC50 = 140 nM T87675 CWG42F 44470318 IC50 = 52 nM T87675 CQEM30 44480711 Ki = 15 nM T87675 CK1Q4M 44481490 Ki = 1550 nM T87675 C8G3YW 44481491 Ki = 1430 nM T87675 C53EDG 44481492 Ki > 800 nM T87675 C4WHX7 44481494 Ki = 45 nM T87675 CRC7Y6 44481495 Ki = 440 nM T87675 C6MCD5 44481764 Ki = 720 nM T87675 CNFT56 44481765 Ki = 280 nM T87675 CRIB07 44481766 Ki = 11 nM T87675 C24AMY 44481768 Ki = 860 nM T87675 C1XA5C 44481769 Ki = 160 nM T87675 C8LN2S 44482036 Ki = 99 nM T87675 CD3YS7 44482037 Ki = 270 nM T87675 C8MEU4 44482038 Ki = 19 nM T87675 CZO5K0 44482039 Ki = 400 nM T87675 CDOZ57 44482040 Ki = 410 nM T87675 CBJ8U7 44482041 Ki = 410 nM T87675 CX5W3P 44482303 Ki = 540 nM T87675 CKS3B9 44482304 Ki = 550 nM T87675 CNZ38Y 44482305 Ki = 15 nM T87675 C1O8SQ 44482306 Ki > 800 nM T87675 CJ56HF 44482307 Ki > 200 nM T87675 CU4N2L 44518360 IC50 = 67 nM T87675 CA1VC7 44518362 IC50 = 786 nM T87675 C8YI9B 44518365 IC50 = 186 nM T87675 C7QU6G 44518503 IC50 = 46 nM T87675 C9GL6Y 44518504 IC50 = 46 nM T87675 CYH6P3 44520205 IC50 < 3 nM T87675 C4H0WR 44520206 IC50 = 88 nM T87675 CP56YC 44520407 IC50 = 171 nM T87675 CG37AY 44520577 IC50 = 37 nM T87675 C9HPB1 44520578 IC50 = 8 nM T87675 C0LY6E 44552561 IC50 = 220 nM T87675 C7KRU3 44552562 IC50 = 170 nM T87675 C97CDF 44555517 IC50 = 484 nM T87675 CY2GA6 44555518 IC50 = 491 nM T87675 CPV8A6 44555519 IC50 = 1376 nM T87675 C9Q8VR 44555761 IC50 = 3168 nM T87675 C68LVU 44555820 IC50 = 372 nM T87675 CP6FY8 44556163 IC50 = 1450 nM T87675 CHA25B 44556214 IC50 = 768 nM T87675 CR2CH3 44556329 IC50 = 750 nM T87675 C3VRO9 44557921 IC50 > 10000 nM T87675 C1A4XG 44562420 IC50 > 10000 nM T87675 C3UV2W 44562431 IC50 > 100000 nM T87675 CC7E4K 44564705 IC50 > 10000 nM T87675 C42ZEW 44564706 IC50 > 10000 nM T87675 C53MCK 44564747 IC50 = 1300 nM T87675 CDI31F 44564748 IC50 > 10000 nM T87675 CA17NT 44564749 IC50 = 1500 nM T87675 CMIZ20 44564750 IC50 > 10000 nM T87675 CSO9F8 44564751 IC50 = 840 nM T87675 C8ATG9 44564787 IC50 = 370 nM T87675 CM50GS 44564788 IC50 = 320 nM T87675 C3Q0DX 44564789 IC50 = 8000 nM T87675 CP40XB 44564790 IC50 > 10000 nM T87675 C35NTB 44564791 IC50 > 10000 nM T87675 CJY83G 44564817 IC50 > 10000 nM T87675 CLK98G 44564818 IC50 > 10000 nM T87675 CF2D1K 44564819 IC50 = 5800 nM T87675 C3CQ9K 44564820 IC50 = 2800 nM T87675 CI8V2L 44564821 IC50 > 10000 nM T87675 C9PO7J 44564860 IC50 > 10000 nM T87675 C16FJW 44564861 IC50 = 4000 nM T87675 C8AMX5 44564862 IC50 = 5700 nM T87675 CTR59U 44564863 IC50 > 10000 nM T87675 C9EY4C 44564864 IC50 > 10000 nM T87675 CG5Z7T 44564910 IC50 > 10000 nM T87675 CU9O4C 44564911 IC50 = 2700 nM T87675 CXZ15S 44564954 IC50 > 10000 nM T87675 CZ78WJ 44564955 IC50 = 6000 nM T87675 CJ1X9V 44565013 IC50 = 160 nM T87675 CN2Q3D 44565014 IC50 = 5500 nM T87675 CM2GN3 44565015 IC50 > 10000 nM T87675 C6RV9I 44565016 IC50 > 10000 nM T87675 CJC85A 44565069 IC50 = 5300 nM T87675 CQ7B2T 44566061 IC50 = 11000 nM T87675 CJG96N 44568212 IC50 = 17000 nM T87675 C3HW7L 44570553 IC50 = 1000 nM T87675 C17PVE 44570554 IC50 = 2000 nM T87675 CLOY92 44570599 IC50 = 3000 nM T87675 CK06LT 44570600 IC50 = 4000 nM T87675 CWFB42 44571820 IC50 > 9500 nM T87675 CAL46Y 44577971 IC50 = 42 nM T87675 CTB96Y 44579918 IC50 = 61 nM T87675 CF32AO 44579957 IC50 = 14340 nM T87675 C07YKU 44579993 IC50 > 100000 nM T87675 C3QLS4 44579994 IC50 > 100000 nM T87675 C6RJZ5 44581565 IC50 = 52 nM T87675 CY6WV9 44591670 IC50 = 182 nM T87675 CG2RT4 44591671 IC50 = 11 nM T87675 C4MJZ5 44591672 IC50 = 4 nM T87675 CO2PF3 44591701 IC50 < 1 nM T87675 CK49WN 45139234 IC50 = 820 nM T87675 C5LNY4 45139425 IC50 > 10000 nM T87675 CW0JQ3 45139426 IC50 > 10000 nM T87675 CA7D0I 45139427 IC50 = 3057 nM T87675 CJ3AQ0 45139428 IC50 = 3839 nM T87675 C21ZAX 45139429 IC50 = 4564 nM T87675 C9SV2P 45139430 IC50 > 10000 nM T87675 CW8A4P 45139609 IC50 = 4050 nM T87675 CY2EH3 45139610 IC50 > 10000 nM T87675 CN15UL 45139611 IC50 = 2312 nM T87675 CX3V6Y 45139612 IC50 = 442 nM T87675 C8DS0B 45139613 IC50 = 6040 nM T87675 CKC91X 45139614 IC50 > 10000 nM T87675 CF3R6G 45139794 IC50 > 10000 nM T87675 CZ9E8D 45139795 IC50 > 10000 nM T87675 CH9QJ8 45139796 IC50 = 1970 nM T87675 CHQ5T2 45139797 IC50 > 10000 nM T87675 CEG96V 45139798 IC50 > 10000 nM T87675 CZ4F0E 45139799 IC50 > 10000 nM T87675 CU3RF1 45139989 IC50 > 10000 nM T87675 CJ0V7H 45139990 IC50 > 10000 nM T87675 CQGZ06 45139991 IC50 = 670 nM T87675 CB6RJ5 45139992 IC50 > 10000 nM T87675 CU5G1L 45139993 IC50 = 4708 nM T87675 CJ46SM 45139994 IC50 > 10000 nM T87675 CI9G7K 45140384 IC50 > 10000 nM T87675 CBH6X7 45141605 IC50 = 1004 nM T87675 CXK9J6 45141799 IC50 = 1144 nM T87675 C3B1OM 45141800 IC50 = 1447 nM T87675 CN94WM 45141801 IC50 = 1688 nM T87675 CLXN28 45141802 IC50 = 672 nM T87675 COM90V 45142011 IC50 = 890 nM T87675 CPO6I5 45142012 IC50 = 2136 nM T87675 CSBG24 45142013 IC50 = 1287 nM T87675 C67GFH 45142014 IC50 = 1923 nM T87675 CZV74M 45142015 IC50 = 2306 nM T87675 CBU5V3 45142016 IC50 = 4643 nM T87675 C0VQ2H 45142243 IC50 > 10000 nM T87675 C2TZO3 45142244 IC50 = 4597 nM T87675 CVA5P9 45142245 IC50 > 10000 nM T87675 C23OLW 45142246 IC50 > 10000 nM T87675 CJ4V3Z 45142247 IC50 > 10000 nM T87675 CH4W1K 45142248 IC50 > 10000 nM T87675 CW3A2T 45142249 IC50 > 10000 nM T87675 CRGD26 45266961 Ki < 3 nM T87675 CY15RC 45267893 Ki = 18 nM T87675 C9UX5Q 45269587 Ki = 3.9 nM T87675 C4W1UX 45269647 IC50 = 213 nM T87675 C87FEM 45270051 IC50 > 40000 nM T87675 CPO6K5 45271266 Ki < 1 nM T87675 C15MIZ 45272990 Ki = 3.9 nM T87675 CU53FK 45273505 IC50 > 40000 nM T87675 CZGB46 46180666 IC50 > 1000 nM T87675 COL3S2 46182728 IC50 <= 4 nM T87675 C8ADR2 46214481 IC50 = 1584.89 nM T87675 CH0ZR1 46214482 IC50 = 3981.07 nM T87675 C2EZU8 46214649 IC50 = 2511.89 nM T87675 C5L1KH 46214650 IC50 > 10000 nM T87675 CRI6G5 46214652 IC50 = 2511.89 nM T87675 CRT51W 46214653 IC50 > 10000 nM T87675 CF57GK 46215462 IC50 = 26 nM T87675 CVW21C 46215644 IC50 = 199.53 nM T87675 CZ58FY 46215814 IC50 = 390 nM T87675 CO9H1K 46215816 IC50 > 10000 nM T87675 CT8G2A 46215988 IC50 = 12589.25 nM T87675 C28SJK 46215992 IC50 = 5011.87 nM T87675 C9JNT0 46216155 IC50 = 199.53 nM T87675 CD96WF 46216494 IC50 = 6309.57 nM T87675 C7NY4T 46223562 IC50 = 42 nM T87675 CG1H6A 46223563 IC50 = 2360 nM T87675 CK4W3S 46223564 IC50 = 92 nM T87675 CGNY46 46223565 IC50 = 169 nM T87675 C0OG3H 46223566 IC50 = 1392 nM T87675 CG18LT 46223796 IC50 > 10000 nM T87675 CEJ1G8 46223797 IC50 = 2848 nM T87675 CU6VF4 46224500 IC50 = 12 nM T87675 CY3HW5 46224684 IC50 = 1100 nM T87675 C1U7IT 46225595 IC50 > 10000 nM T87675 C8YPN0 46225596 IC50 = 230 nM T87675 C34JTS 46225597 IC50 = 65 nM T87675 CGD73B 46225598 IC50 = 290 nM T87675 C3E0PU 46225599 IC50 = 390 nM T87675 CRDY89 46225610 IC50 = 27 nM T87675 C0JMT8 46225611 IC50 = 62 nM T87675 CF0D5J 46225612 IC50 = 14 nM T87675 CFVO38 46225632 IC50 = 200 nM T87675 CLZ1O6 46225634 IC50 = 26 nM T87675 C07VDX 46225635 IC50 = 110 nM T87675 CT70DX 46225640 IC50 = 230 nM T87675 CJUF68 46225641 IC50 = 690 nM T87675 C6AJ5N 46225647 IC50 = 26 nM T87675 C2WCV1 46225648 IC50 = 400 nM T87675 CBS96A 46225649 IC50 = 1200 nM T87675 C38BFC 46225657 IC50 = 120 nM T87675 CD0A6F 46225658 IC50 = 9400 nM T87675 C1B3KS 46225663 IC50 = 9 nM T87675 CU46XI 46225664 IC50 = 54 nM T87675 CO3HS2 46225665 IC50 = 24 nM T87675 C2UV1S 46225666 IC50 = 60 nM T87675 CX5B1G 46225667 IC50 = 85 nM T87675 C2Q9OH 46225668 IC50 = 3300 nM T87675 C16LEO 46225679 IC50 > 10000 nM T87675 CM14FH 46225680 IC50 = 800 nM T87675 CQS96E 46225681 IC50 = 1300 nM T87675 CJIK35 46225682 IC50 = 1600 nM T87675 C8S4QA 46225688 IC50 = 340 nM T87675 CYT37A 46232443 IC50 > 50000 nM T87675 C48ZVW 46232555 IC50 = 6400 nM T87675 CS9B1U 46232556 IC50 = 22000 nM T87675 CC2WT4 46232590 IC50 = 3500 nM T87675 CXR70F 46233220 IC50 = 1308 nM T87675 CH6V1G 46233221 IC50 > 10000 nM T87675 CAU1C9 46233286 IC50 = 1237 nM T87675 C7ON5A 46233287 IC50 = 3500 nM T87675 CJE67S 46233288 IC50 = 1288 nM T87675 CBF4Z6 46233289 IC50 = 3112 nM T87675 C1IZ5P 46236622 IC50 = 197 nM T87675 CW7F4D 46236768 IC50 = 228 nM T87675 CCSD82 46236769 IC50 = 203 nM T87675 CF2W4N 46237019 IC50 = 1701 nM T87675 C97VFZ 46237140 IC50 = 2819 nM T87675 CKTI63 46237141 IC50 = 5477 nM T87675 CS35CW 46237142 IC50 = 579 nM T87675 CCZ65K 46237143 IC50 = 2445 nM T87675 C2MRG9 46240951 IC50 > 10000 nM T87675 C3OQ6X 46700767 IC50 = 178 nM T87675 CGO1J5 46830766 Ki = 18 nM T87675 CF7HK2 46830767 Ki = 31 nM T87675 C2HJ1X 46830768 Ki = 7.6 nM T87675 C79BLH 46846452 IC50 = 362 nM T87675 CK2ZQ4 46846637 IC50 = 271 nM T87675 CP1XL3 46846638 IC50 = 7 nM T87675 C17MQN 46846639 IC50 = 29 nM T87675 C5NH7Q 46846640 IC50 = 61 nM T87675 CF6L2A 46846641 IC50 = 8 nM T87675 C5TJ2U 46846734 IC50 = 14 nM T87675 CB5Z6C 46846735 IC50 = 21 nM T87675 CQWL17 46846948 IC50 = 63 nM T87675 CK6XQ9 46846949 IC50 = 208 nM T87675 CJ05RO 46846951 IC50 = 210 nM T87675 CEBI80 46846952 IC50 = 357 nM T87675 C08JXQ 46846953 IC50 = 724 nM T87675 C2RGP1 46847064 IC50 = 31 nM T87675 C5PA2R 46847066 IC50 = 560 nM T87675 CD65VE 46847181 IC50 = 443 nM T87675 C7NUY3 46847552 IC50 = 84 nM T87675 C2MO3J 46847553 IC50 = 252 nM T87675 CTFH14 46847557 IC50 = 57 nM T87675 CF19AB 46847648 IC50 = 34 nM T87675 CCV16U 46847847 IC50 = 12 nM T87675 C8G6BZ 46847848 IC50 = 1780 nM T87675 C82FUA 46847849 IC50 = 1980 nM T87675 C4QU6W 46854745 IC50 = 304 nM T87675 CO58XV 46854746 IC50 = 5831 nM T87675 C9MS1U 46854890 IC50 > 10000 nM T87675 CT8AF6 46854894 IC50 = 807 nM T87675 CUE7V1 46855041 IC50 = 296 nM T87675 CO9T8Q 46855042 IC50 = 796 nM T87675 C6JYX5 46855043 IC50 = 640 nM T87675 CV4NU2 46855044 IC50 = 792 nM T87675 CM8RW2 46855045 IC50 = 760 nM T87675 CLEX76 46855046 IC50 = 535 nM T87675 COQ2S4 46855195 IC50 = 827 nM T87675 CEY4R9 46855196 IC50 = 334 nM T87675 C0KU4M 46855197 IC50 = 640 nM T87675 C1BW5G 46855198 IC50 = 973 nM T87675 C63YRO 46855199 IC50 = 945 nM T87675 CXA1H4 46866784 IC50 = 9 nM T87675 C8WT0Y 46866785 IC50 = 8 nM T87675 CFL32P 46866786 IC50 = 40 nM T87675 CIBN38 46866787 IC50 = 650 nM T87675 CB2P8Q 46866788 IC50 = 17 nM T87675 C8J5QY 46866895 IC50 = 32 nM T87675 CEN91W 46866896 IC50 = 4 nM T87675 CTW3P1 46866897 IC50 = 5 nM T87675 C9F1GJ 46866898 IC50 = 6 nM T87675 C74EKS 46867015 IC50 = 30 nM T87675 C4B0FJ 46867016 IC50 = 6 nM T87675 CK1Y3J 46867128 IC50 = 2 nM T87675 CB92AK 46867805 IC50 = 50 nM T87675 CLU9A0 46867945 IC50 = 81 nM T87675 CXO3G4 46867947 IC50 = 16 nM T87675 C2XL0N 46867948 IC50 = 81 nM T87675 CY6Q1P 46867949 IC50 = 52 nM T87675 C65FYN 46868083 IC50 = 3 nM T87675 CJA45H 46868085 IC50 = 29 nM T87675 CZQ57K 46868086 IC50 = 10 nM T87675 CJL9N7 46868087 IC50 = 10 nM T87675 C1EIB5 46868212 IC50 = 3 nM T87675 CX8V7J 46868352 IC50 = 115 nM T87675 C9SGR3 46868503 IC50 = 118 nM T87675 CHMW94 46868504 IC50 = 75 nM T87675 C6AM4H 46868505 IC50 = 277 nM T87675 C5G0WX 46868506 IC50 = 178 nM T87675 CS03JT 46868507 IC50 = 258 nM T87675 C2Y6AZ 46868508 IC50 = 210 nM T87675 C49DEU 46868647 IC50 = 55 nM T87675 C4NGQ3 46868648 IC50 = 79 nM T87675 C6SMX9 46868649 IC50 = 55 nM T87675 C5VZA4 46868651 IC50 = 9 nM T87675 CLS29B 46872626 IC50 > 10000 nM T87675 CT48CR 46883054 IC50 = 1400 nM T87675 C9ZVS1 46883055 IC50 = 490 nM T87675 C5ETX6 46883135 IC50 = 40 nM T87675 CVG27D 46883136 IC50 = 28 nM T87675 CCQ6N9 46883137 IC50 = 64 nM T87675 CR48QI 46883180 IC50 = 17 nM T87675 C5EM0A 46883181 IC50 = 20 nM T87675 CRE96X 46885625 IC50 = 631 nM T87675 CZRY30 46885675 IC50 > 10000 nM T87675 C2U8YW 46886303 IC50 = 1700 nM T87675 CTOQ14 46886304 IC50 = 22 nM T87675 C86YZR 46886305 IC50 = 19 nM T87675 C2O8RZ 46886323 IC50 = 65 nM T87675 CRAD15 46886342 IC50 = 17 nM T87675 CNJ50M 46886343 IC50 = 240 nM T87675 CP4O2N 46886344 IC50 = 160 nM T87675 CHL2F0 46886392 IC50 = 42 nM T87675 CKIH05 46886393 IC50 = 35 nM T87675 CMH09O 46886394 IC50 = 280 nM T87675 CQ6A0O 46886395 IC50 = 350 nM T87675 C5M8UY 46886877 IC50 > 10000 nM T87675 C6XIZ3 46886878 IC50 > 10000 nM T87675 CQI12F 46886956 IC50 = 270 nM T87675 C3RIH2 46886957 IC50 > 10000 nM T87675 CZ4J8I 46886958 IC50 = 176 nM T87675 CBJ26E 46886959 IC50 = 116 nM T87675 CMU45C 46886960 IC50 = 607 nM T87675 C38MVY 46887029 IC50 = 158 nM T87675 C3Y5NA 46887030 IC50 = 128 nM T87675 C1SJ7I 46887031 IC50 > 10000 nM T87675 C32MST 46887032 IC50 > 10000 nM T87675 CN4O5T 46887033 IC50 > 10000 nM T87675 C7JG4Q 46887069 IC50 > 10000 nM T87675 CYG3B2 46887070 IC50 = 1181 nM T87675 C82SLV 46887071 IC50 > 10000 nM T87675 CD4Y9O 46887101 IC50 > 10000 nM T87675 CYL4K8 46887102 IC50 > 10000 nM T87675 C29OLT 46887103 IC50 > 10000 nM T87675 CW5P4R 46887104 IC50 > 10000 nM T87675 C1W3QP 46887105 IC50 > 10000 nM T87675 CJ0QH7 46887137 IC50 > 10000 nM T87675 C8GO5N 46887138 IC50 > 10000 nM T87675 CL5IQ9 46887139 IC50 > 10000 nM T87675 CFV71W 46887140 IC50 > 10000 nM T87675 C45OAG 46887187 IC50 = 2497 nM T87675 CW13FN 46887188 IC50 > 10000 nM T87675 C5X8BP 46887189 IC50 > 10000 nM T87675 CB8Q1F 46887190 IC50 > 10000 nM T87675 CK1YB8 46887222 IC50 > 10000 nM T87675 CT80IX 46888385 IC50 = 5111 nM T87675 CEG84F 46888585 IC50 = 3848 nM T87675 C38XJC 46888586 IC50 = 5600 nM T87675 CE59WH 46888607 IC50 = 5770 nM T87675 CE3N4O 46888608 IC50 = 8156 nM T87675 CY48GN 46888609 IC50 = 2150 nM T87675 CJ34VB 46888641 IC50 = 792 nM T87675 C4A9KL 46888642 IC50 = 377 nM T87675 CIG2O5 46888643 IC50 = 969 nM T87675 CA8X6N 46888676 IC50 = 5676 nM T87675 CZN1S5 46888677 IC50 = 3392 nM T87675 CYG5P0 46888678 IC50 = 6810 nM T87675 CV6BH4 46888679 IC50 = 126 nM T87675 CDFP47 46888680 IC50 = 62 nM T87675 CB39WR 46888681 IC50 = 113 nM T87675 CHEB15 46888682 IC50 = 45 nM T87675 C7KM8F 46888683 IC50 = 42 nM T87675 C1SBV8 46888684 IC50 = 22 nM T87675 C2X3KJ 46888685 IC50 = 94 nM T87675 C53EWU 46888686 IC50 = 59 nM T87675 CW7C4L 46888746 IC50 = 58 nM T87675 C5RI8V 46888747 IC50 = 366 nM T87675 CXW80O 46888771 IC50 = 42 nM T87675 C0KN5S 46888772 IC50 = 70 nM T87675 CIN2Q6 46888773 IC50 = 23 nM T87675 C1O9ES 46888774 IC50 = 250 nM T87675 C98GDK 46889922 IC50 = 10 nM T87675 CX18GT 46889932 IC50 = 15 nM T87675 CM12LB 46889933 IC50 = 10 nM T87675 CEH68I 46889934 IC50 = 3 nM T87675 CONK89 46889935 IC50 = 10 nM T87675 CM02UJ 46890253 IC50 = 332 nM T87675 CB7VI8 46890254 IC50 = 1658 nM T87675 C7V3IA 46890314 IC50 = 225 nM T87675 CHE6A1 46890315 IC50 = 534 nM T87675 CTZ71Y 46898039 IC50 = 2.09 nM T87675 C5G2VE 46909588 IC50 > 10000 nM T87675 CL0O4U 46911726 Ki = 1.2 nM T87675 CVHG53 46913876 IC50 = 563 nM T87675 CJ0M3S 46913877 IC50 = 2170 nM T87675 CQLT07 46913878 IC50 = 2190 nM T87675 C8Z1VS 46913879 IC50 = 2450 nM T87675 CMVA69 46913880 IC50 = 2270 nM T87675 CEC9O6 46914012 IC50 = 2340 nM T87675 C5L9YG 46914302 IC50 = 456 nM T87675 C1H5QN 46915919 IC50 = 720 nM T87675 CR01PN 46915920 IC50 = 39 nM T87675 CJXV84 46916061 IC50 = 218 nM T87675 CS68OQ 46916062 IC50 = 281 nM T87675 CFE0B3 46916063 IC50 = 117 nM T87675 CCN08S 46934144 IC50 > 100000 nM T87675 CV4X7L 49787166 IC50 = 75 nM T87675 CCSP59 49800150 IC50 = 190 nM T87675 CY3EO0 49800670 IC50 = 17 nM T87675 CHSF07 49806372 IC50 > 1000 nM T87675 C5ME3S 49806721 IC50 > 50000 nM T87675 CF91RS 49843531 IC50 > 10000 nM T87675 C7A6IZ 49850211 IC50 = 30 nM T87675 CA4QJ0 49867401 IC50 <= 4 nM T87675 CYKC34 50898605 IC50 = 212 nM T87675 CA06SB 50898682 IC50 = 195 nM T87675 CU2WV0 50898683 IC50 = 78 nM T87675 C6IHC3 50898684 IC50 = 143 nM T87675 C1FL0P 50898685 IC50 = 128 nM T87675 CP4CI5 50898686 IC50 = 564 nM T87675 CCS4B1 50898764 IC50 = 193 nM T87675 C5J2WG 50898765 IC50 = 202 nM T87675 C3MFH7 50898766 IC50 = 103 nM T87675 CU9K2Q 50898767 IC50 = 115 nM T87675 CX3J2C 50898768 IC50 = 123 nM T87675 CMG3J8 50898859 IC50 = 796 nM T87675 CK5TH3 50906783 IC50 = 270 nM T87675 CD2K4R 50908681 Ki > 1000000 nM T87675 CRCT70 50909914 IC50 = 1258.93 nM T87675 C0XDI4 50909915 IC50 = 1258.93 nM T87675 CUJL92 50909916 IC50 = 501.19 nM T87675 C51DKX 50909917 IC50 = 398.11 nM T87675 C2Y6QS 50938552 IC50 > 10000 nM T87675 CVTS82 50993809 IC50 = 14000 nM T87675 C8IL9F 50994667 IC50 <= 4 nM T87675 C4QA8D 50994668 IC50 <= 4 nM T87675 CR0B8X 50994669 IC50 <= 4 nM T87675 C9UK6T 50994670 IC50 <= 4 nM T87675 CIF3W1 50994671 IC50 <= 4 nM T87675 CAZQ43 51003133 IC50 <= 4 nM T87675 C9NYP4 51036677 IC50 > 10000 nM T87675 C4WRY3 51037112 IC50 > 10000 nM T87675 CRI28Z 51037948 IC50 > 10000 nM T87675 CYD4A2 51354035 IC50 = 7943.28 nM T87675 CW2T3N 51354036 IC50 > 10000 nM T87675 CH8NX6 51354037 IC50 > 10000 nM T87675 CK63DI 51354327 IC50 = 1258.93 nM T87675 CC6PZ4 51354328 IC50 = 1258.93 nM T87675 C2FVX4 51354329 IC50 = 1995.26 nM T87675 CV06QD 51354330 IC50 = 6309.57 nM T87675 CR3AC1 51354331 IC50 = 1584.89 nM T87675 CUXD62 51354613 IC50 = 63.1 nM T87675 C3G1VK 51354899 IC50 > 10000 nM T87675 CK7NP1 51354900 IC50 > 10000 nM T87675 CEDN75 51354901 IC50 > 10000 nM T87675 CB0EU1 51355190 IC50 = 7943.28 nM T87675 CYZ03E 51356852 IC50 = 3162.28 nM T87675 CL3S8F 51356853 IC50 = 3162.28 nM T87675 C67DUF 51356854 IC50 = 1995.26 nM T87675 CAU2F6 51356855 IC50 > 10000 nM T87675 CD07RV 51356856 IC50 > 10000 nM T87675 CFM5I7 51357137 IC50 = 12589.25 nM T87675 CP6R5J 51357138 IC50 > 10000 nM T87675 CWCJ29 51357417 IC50 = 7943.28 nM T87675 CS9WE1 51357418 IC50 > 10000 nM T87675 C5G7BY 51357419 IC50 > 10000 nM T87675 CBM4P9 51357696 IC50 > 10000 nM T87675 C65MXB 51357954 IC50 = 5011.87 nM T87675 CXA03W 52920796 IC50 <= 4 nM T87675 C1VML8 52936434 Ki = 2600 nM T87675 CEQN27 52936621 Ki > 1000 nM T87675 CM24LF 52938983 IC50 < 1 nM T87675 C2UH4P 52940893 IC50 <= 4 nM T87675 CQB32I 52941003 IC50 <= 4 nM T87675 CC42PX 52942070 IC50 <= 4 nM T87675 C38PKY 52942116 IC50 <= 4 nM T87675 C31EGF 52942164 IC50 <= 4 nM T87675 CF1X3D 52942218 IC50 <= 4 nM T87675 C15XBH 52942244 IC50 <= 4 nM T87675 CYO6V1 52943688 IC50 = 6700 nM T87675 CX25YN 52943772 IC50 = 3750 nM T87675 CDXB91 52943898 IC50 = 208 nM T87675 C7T8NP 52944489 IC50 <= 4 nM T87675 C2L5VS 52944583 IC50 = 7310 nM T87675 C5A1IX 52944643 IC50 <= 4 nM T87675 C93RQV 52944679 IC50 <= 4 nM T87675 CIL69W 52944937 IC50 = 2900 nM T87675 CPCI51 52944938 IC50 = 2500 nM T87675 C1LY7R 52945074 IC50 = 4500 nM T87675 CN0AS2 52945317 IC50 = 9700 nM T87675 C7EWH2 52945730 IC50 <= 4 nM T87675 C8MCU4 52945733 IC50 <= 4 nM T87675 C34WPX 52945791 IC50 <= 4 nM T87675 CM90HV 52946216 IC50 = 7900 nM T87675 CD3F7J 52946403 IC50 = 18 nM T87675 CIM9A5 52946956 IC50 <= 4 nM T87675 C0OAD7 52947107 IC50 <= 4 nM T87675 CRL93S 52947958 IC50 > 10000 nM T87675 C0CJD8 52948167 IC50 <= 4 nM T87675 CRFY84 52948208 IC50 <= 4 nM T87675 CKSH24 52948244 IC50 <= 4 nM T87675 C8FMO5 52948247 IC50 = 45 nM T87675 CZ19SU 52948345 IC50 <= 4 nM T87675 C17DLE 52948743 IC50 = 105 nM T87675 CMV3N5 52948942 IC50 = 7200 nM T87675 CQ3H5Y 52948987 IC50 = 44 nM T87675 CF8WT5 52949399 IC50 <= 4 nM T87675 CE5M0X 52949491 IC50 = 5480 nM T87675 C42QAS 52949563 IC50 <= 4 nM T87675 C9J3GU 52949936 IC50 = 6700 nM T87675 CYN1Q6 52949977 IC50 = 152 nM T87675 C0TOX3 52949997 IC50 = 4200 nM T87675 C7UT2K 52950167 IC50 = 5500 nM T87675 C7QNV0 53308639 IC50 = 180 nM T87675 CD35QU 53308640 IC50 = 17 nM T87675 C7LRW4 53316508 IC50 = 277 nM T87675 CONY06 53316509 IC50 = 4400 nM T87675 CV6TO2 53317837 IC50 = 5 nM T87675 CE8OY2 53317913 IC50 <= 4 nM T87675 CS6O1B 53318071 IC50 = 11940 nM T87675 C24GBF 53319075 IC50 = 4.8 nM T87675 CEL08W 53320550 IC50 <= 4 nM T87675 CB4C2H 53320716 IC50 = 0.5 nM T87675 CNT63V 53321767 IC50 = 14 nM T87675 C94EAD 53322007 IC50 > 100000 nM T87675 C2W9OA 53324451 IC50 > 10000 nM T87675 C1VOB5 53325994 IC50 = 86150 nM T87675 CNPM14 53341082 IC50 > 3000 nM T87675 C0SWH5 53348216 IC50 > 40000 nM T87675 CM7P3W 53357328 IC50 > 50000 nM T87675 CE8OA7 53357593 IC50 = 290 nM T87675 C1CR6S 53363307 IC50 > 10000 nM T87675 CK03PA 53363389 IC50 > 10000 nM T87675 C8NA4L 53384644 IC50 > 30000 nM T87675 C71OXL 53388145 IC50 = 4800000 nM T87675 CDL28G 53388146 IC50 > 100000000 nM T87675 C7KM5B 53388319 IC50 = 14 nM T87675 CVG90B 53389651 IC50 > 10000 nM T87675 CX5G1Z 54580622 Ki = 20 nM T87675 CD8UO5 54580769 Ki = 9.7 nM T87675 CRN28X 54581311 IC50 = 125.89 nM T87675 CN7Z6J 54581629 Ki = 4.5 nM T87675 C31NWF 54581705 Ki = 310 nM T87675 CO9QV2 54582429 IC50 = 12000 nM T87675 C7UZ0J 54583660 Ki = 3.8 nM T87675 C6XC1V 54585332 IC50 = 4800 nM T87675 C6H7VA 54585578 Ki = 5.3 nM T87675 C7W9PB 54585645 Ki = 66 nM T87675 CFG1L6 54586483 Ki = 28 nM T87675 CN5WJ3 54586639 Ki = 2.3 nM T87675 CXYV09 54587513 Ki = 8.5 nM T87675 CE1ZK6 54759168 IC50 > 10000 nM T87675 CY3V6S 54764326 IC50 > 10000 nM T87675 C0H9PE 54768609 IC50 = 101 nM T87675 C23GVF 54768644 IC50 = 104 nM T87675 CC6G4T 54768645 IC50 = 9238 nM T87675 CG76TH 56587958 IC50 = 8.9 nM T87675 CN1E6U 56587959 IC50 = 0.74 nM T87675 CK7QZ5 56587961 IC50 = 3.7 nM T87675 CM13KI 56587962 IC50 = 149 nM T87675 C53YRZ 56587963 IC50 = 35.1 nM T87675 C6R7CI 56587964 IC50 = 2.1 nM T87675 C2SG7Y 56587965 IC50 = 43 nM T87675 C83VCG 56587966 IC50 = 0.2 nM T87675 C67EBW 56587967 IC50 = 3.1 nM T87675 CD2U6K 56587968 IC50 = 28 nM T87675 C5KR6N 56595558 Ki = 103 nM T87675 COI9U2 56595687 Ki > 7000 nM T87675 C2AM6B 56595688 Ki = 2000 nM T87675 CFY2I4 56595689 Ki > 4000 nM T87675 CAM8E1 56595690 Ki > 3000 nM T87675 CN5EV7 56595691 Ki > 2500 nM T87675 C6ET0W 56595693 Ki = 2100 nM T87675 CM8JX1 56604907 IC50 = 1000 nM T87675 CN9QD7 56643097 IC50 > 10000 nM T87675 C0R5FU 56658064 IC50 > 10000 nM T87675 CTR10F 56658543 Ki = 2600 nM T87675 CXIZ08 56659726 IC50 > 10000 nM T87675 C8IZ4J 56659759 IC50 = 680 nM T87675 CPG0I4 56659823 IC50 > 1000 nM T87675 C4UPH5 56659824 IC50 = 1170 nM T87675 CVDT38 56659825 IC50 > 1000000 nM T87675 CUV7W2 56661575 IC50 = 5 nM T87675 CWV3Y1 56661576 IC50 = 150 nM T87675 CXCY28 56662867 IC50 = 8 nM T87675 CC90EV 56662926 IC50 = 46 nM T87675 CB3Q1P 56663194 IC50 > 10000 nM T87675 C3A7HL 56663233 IC50 = 540 nM T87675 CY12ML 56663288 IC50 = 4990 nM T87675 CK53GA 56663289 IC50 = 850 nM T87675 CY2RD1 56663290 IC50 > 1000 nM T87675 CC4IM3 56664990 IC50 = 30 nM T87675 CP4B3L 56666399 IC50 = 6 nM T87675 CK75JI 56666400 IC50 = 50 nM T87675 CO6N5S 56666401 IC50 = 83 nM T87675 C2JRW4 56666402 IC50 = 82 nM T87675 CZYH57 56666592 IC50 = 152 nM T87675 C6XVT5 56666663 IC50 = 170 nM T87675 CKE5U3 56666717 IC50 = 220 nM T87675 C28LZS 56668430 IC50 = 6 nM T87675 CIM94L 56668847 IC50 > 100000000 nM T87675 C8L2VE 56669813 IC50 = 3700 nM T87675 C3C1XF 56669814 IC50 = 81 nM T87675 C9FR3E 56669815 IC50 = 27 nM T87675 C1HTO5 56670140 IC50 = 1640 nM T87675 CI0JY1 56671940 IC50 = 350 nM T87675 CTJ5B4 56672286 IC50 = 13 nM T87675 CCSO01 56673303 IC50 > 10000 nM T87675 CHEK09 56673306 IC50 = 30 nM T87675 CC3J1A 56673651 IC50 = 340 nM T87675 C4TD2Q 56673654 IC50 = 1710 nM T87675 CVBU67 56675317 IC50 = 20 nM T87675 CY43DK 56675318 IC50 = 110 nM T87675 C8PK0W 56675716 IC50 > 100000000 nM T87675 C2XE7T 56676636 IC50 = 603 nM T87675 C2BL7S 56676833 IC50 = 677 nM T87675 CS3EP0 56676834 IC50 > 10000 nM T87675 CRG16Y 56676835 IC50 = 1376 nM T87675 C6B1PU 56676891 IC50 > 10000 nM T87675 CGN54D 56676922 IC50 > 1000000 nM T87675 CU0M8W 56676973 IC50 = 430 nM T87675 CUD53B 56676975 IC50 = 390 nM T87675 CO2GI9 56676977 IC50 > 1000000 nM T87675 CM0TN3 56678661 IC50 = 5 nM T87675 CG0Y7I 56678662 IC50 = 9 nM T87675 CLW54U 56678663 IC50 = 260 nM T87675 CO9P6E 56679965 IC50 = 170 nM T87675 C1GC5S 56679966 IC50 <= 4 nM T87675 CFVN60 56679967 IC50 = 14 nM T87675 CFS43O 56680303 IC50 > 1000 nM T87675 C5RK1U 56680304 IC50 > 1000 nM T87675 CG1WU4 56681977 IC50 = 95 nM T87675 C1KJD9 56683295 IC50 = 17 nM T87675 CSX3Y4 56683569 IC50 > 1000000 nM T87675 CVM7U4 56683624 IC50 > 1000 nM T87675 C4Z0OC 56834890 IC50 = 140 nM T87675 C67TJQ 56834891 IC50 = 460 nM T87675 CR50TJ 56835147 IC50 = 2680 nM T87675 CI5ZJ7 56835161 IC50 > 100000 nM T87675 CJBL48 56925034 IC50 = 444 nM T87675 CIV57W 56947168 IC50 = 8810 nM T87675 CR16SD 56947170 IC50 = 4940 nM T87675 CP8J4Y 56973724 IC50 = 21000 nM T87675 CPJX47 57111159 Ki = 76300 nM T87675 C5YRF8 57328039 IC50 = 4 nM T87675 CP7UB8 57383477 IC50 = 28 nM T87675 CM61IS 57384257 IC50 = 1 nM T87675 C8OL3E 57384510 IC50 = 2 nM T87675 CACW05 57386803 IC50 = 7930 nM T87675 CG14VM 57387301 IC50 = 2330 nM T87675 CH53XJ 57391650 IC50 > 10000 nM T87675 CF4U0R 57391651 IC50 > 10000 nM T87675 CE8T5V 57393795 IC50 > 20000 nM T87675 CFM9W7 57394672 IC50 = 91000 nM T87675 CG8FR3 57394673 IC50 = 7000 nM T87675 C73BDI 57394674 IC50 = 6000 nM T87675 C8W6IG 57395117 IC50 > 30000 nM T87675 CRLG52 57395119 IC50 > 10000 nM T87675 CX6GJ7 57396885 IC50 > 10000 nM T87675 CU2PF5 57398440 IC50 = 6195 nM T87675 C59OYH 57398540 IC50 > 10000 nM T87675 CG4D3H 57398639 IC50 > 10000 nM T87675 CS68OM 57399870 IC50 = 242000 nM T87675 CR81YF 57399871 IC50 = 137000 nM T87675 CMQ7A6 57400314 IC50 > 10000 nM T87675 C67BJY 57401650 IC50 = 234000 nM T87675 C8H2MA 57402115 IC50 > 10000 nM T87675 CEG5Q7 57403865 IC50 > 10000 nM T87675 CK7L8O 57403866 IC50 > 10000 nM T87675 CZSM95 57412684 IC50 = 1500 nM T87675 CE59QS 57505507 IC50 = 360 nM T87675 CEW5L7 57522817 IC50 = 30000 nM T87675 C4SEH5 57522818 IC50 = 30000 nM T87675 CF8IP6 57522819 IC50 > 100000 nM T87675 CJ56CE 57522820 IC50 = 5000 nM T87675 C3XI2P 57523093 IC50 = 30000 nM T87675 CUH3B5 57523094 IC50 > 100000 nM T87675 C3QF2X 57523095 IC50 > 100000 nM T87675 C68VTP 57946373 IC50 = 41 nM T87675 C78UXM 57946415 IC50 = 20 nM T87675 CP2S6W 57946419 IC50 = 61 nM T87675 CEA28W 57946425 IC50 = 342 nM T87675 CAJ4N9 57946484 IC50 = 123 nM T87675 C3EA1I 57946503 IC50 > 10000 nM T87675 CWL0A1 57946504 IC50 = 98.3 nM T87675 C2N3RC 57946511 IC50 = 160 nM T87675 CCY9J3 57946541 IC50 = 203 nM T87675 CQJO89 57946544 IC50 = 141 nM T87675 C8KCF9 57946556 IC50 = 50 nM T87675 C3CXL6 57946584 IC50 > 10000 nM T87675 C6YJG0 57946585 IC50 = 929 nM T87675 C2CJM6 57946594 IC50 = 367 nM T87675 C2L5MZ 57946607 IC50 = 80 nM T87675 CD6ZP3 58009815 IC50 = 570 nM T87675 CWU1Y3 58009825 IC50 = 340 nM T87675 C8S6MY 58010054 IC50 = 130 nM T87675 CM1B4V 58010265 IC50 = 40 nM T87675 CVK0G4 58056356 IC50 = 42000 nM T87675 CI50KU 58167984 IC50 = 0.3 nM T87675 CM2ZN1 58167992 IC50 = 1030 nM T87675 CL9P3V 58168008 IC50 = 3010 nM T87675 C87VTG 58168047 IC50 = 1150 nM T87675 C6LQ3W 58168051 IC50 = 7 nM T87675 C6F3DH 58168083 IC50 = 615 nM T87675 CBU03C 58168094 IC50 = 27 nM T87675 CQK0L7 58168151 IC50 = 7 nM T87675 C3R6DT 58168169 IC50 = 7 nM T87675 CMR59F 58282865 IC50 < 4 nM T87675 CI37CQ 58394927 IC50 = 640 nM T87675 C6KO0G 58395044 IC50 = 740 nM T87675 C2I3QW 58486157 IC50 > 1000 nM T87675 C7ZKF5 58486186 IC50 > 1000 nM T87675 CBF7L4 58486208 IC50 > 1000 nM T87675 CM91GS 58486210 IC50 > 1000 nM T87675 CQPU86 58486223 IC50 > 1000 nM T87675 C51FBH 58486335 IC50 > 1000 nM T87675 CB42EF 58557147 IC50 = 3200 nM T87675 C8X6YE 58557497 IC50 = 4300 nM T87675 CQTB49 58692572 Ki > 100000 nM T87675 CZ3TG1 59375154 IC50 > 2000 nM T87675 CL6Q5B 59503456 IC50 = 21 nM T87675 CV7N4L 59503457 IC50 = 168 nM T87675 CT15SY 59503468 IC50 = 753 nM T87675 CN8A1T 59503488 IC50 = 239 nM T87675 C4TQG5 59503510 IC50 = 102 nM T87675 C6OP8J 59503511 IC50 > 3000 nM T87675 CK36AN 59503540 IC50 = 22 nM T87675 CKSV12 59503547 IC50 = 340 nM T87675 CE4C9L 59503584 IC50 > 3000 nM T87675 CWB60P 59503611 IC50 = 1567 nM T87675 CVLR79 59503615 IC50 = 213 nM T87675 CAC9V1 59503633 IC50 = 100 nM T87675 CHPZ79 59503635 IC50 > 3000 nM T87675 CT47FC 59503644 IC50 = 18 nM T87675 C1KYO9 59503657 IC50 = 1627 nM T87675 CP9A8T 59503659 IC50 < 4 nM T87675 C05AKO 59503686 IC50 = 53 nM T87675 C2MO0R 59503688 IC50 = 40 nM T87675 CM3TJ8 59503701 IC50 = 1803 nM T87675 CRM90T 59503709 IC50 = 34 nM T87675 C1MA6J 59503711 IC50 = 122 nM T87675 C4P7KI 59503724 IC50 > 3000 nM T87675 CY4VQ0 59503725 IC50 = 1223 nM T87675 CHE68K 59503732 IC50 = 198 nM T87675 CX29EU 59503744 IC50 = 27 nM T87675 C6CJU5 59503756 IC50 = 30 nM T87675 C2SW7U 59503836 IC50 = 45 nM T87675 CRIW40 59825670 IC50 > 10000 nM T87675 C63REN 59825673 IC50 = 4 nM T87675 C3UW1D 59825681 IC50 = 22 nM T87675 CI4F9C 59825699 IC50 = 31 nM T87675 C9LWV7 59825704 IC50 = 22 nM T87675 CO34FC 59825742 IC50 = 3 nM T87675 C65BUA 59825756 IC50 = 15 nM T87675 C3ZSR4 59825772 IC50 = 34 nM T87675 CI8C9G 59825774 IC50 = 8 nM T87675 CZ8S5M 59825775 IC50 = 10 nM T87675 COH62U 60097413 IC50 > 5000 nM T87675 C1MR8Q 60097495 IC50 > 1000 nM T87675 CW78PN 60138156 IC50 = 38.2 nM T87675 CDAG83 60168111 IC50 = 160 nM T87675 C08VMZ 60198892 IC50 = 73 nM T87675 C4K8YJ 60198895 IC50 = 25 nM T87675 C5ZB2G 60199003 IC50 = 490 nM T87675 CN3W2C 60199004 IC50 > 1000 nM T87675 CTR58Y 60199005 IC50 = 38 nM T87675 C5VY6S 66546721 IC50 > 100000 nM T87675 CMT23K 66546905 IC50 > 100000 nM T87675 C2HO8D 66547424 IC50 = 17000 nM T87675 CJ5HI6 66547425 IC50 > 40000 nM T87675 CLWU09 66547597 IC50 > 100000 nM T87675 C6SFP7 66547759 IC50 = 53000 nM T87675 CM4PW9 66548104 IC50 = 75000 nM T87675 C8ZJF7 66548458 IC50 > 40000 nM T87675 CZ0KN3 66548460 IC50 > 100000 nM T87675 CGW4L5 66548650 IC50 > 100000 nM T87675 C7Q2CM 66548653 IC50 > 40000 nM T87675 CI41NJ 66548849 IC50 = 3200 nM T87675 CTJ64B 66548850 IC50 = 8500 nM T87675 CK6WO0 66552478 IC50 < 10000 nM T87675 C7MD5X 66556536 IC50 = 1258.93 nM T87675 CK0XR7 66560844 IC50 = 2 nM T87675 C79HET 66721774 IC50 = 1279 nM T87675 C1HSE0 67035086 IC50 = 3100 nM T87675 CWI6K5 67035106 IC50 > 10000 nM T87675 C38RGB 67035556 IC50 > 10000 nM T87675 CVT35R 67097557 Ki = 4 nM T87675 CSQ3J1 67098421 Ki = 29 nM T87675 CJV8O4 67098558 Ki = 10 nM T87675 CE49GC 67098566 Ki = 4 nM T87675 COD28B 67098794 Ki = 6 nM T87675 C23QPJ 67098846 Ki < 1 nM T87675 C13OVI 67098869 Ki = 6 nM T87675 C9KQT3 67098926 Ki = 2 nM T87675 C52XBW 67098971 Ki = 1 nM T87675 C37NKO 67129970 IC50 > 10000 nM T87675 CK80LJ 67130050 IC50 > 10000 nM T87675 CV63UL 67240318 IC50 > 10000 nM T87675 CUI07E 67378360 IC50 = 75 nM T87675 C6D3QJ 67448476 IC50 > 1000 nM T87675 C7N4ZS 68034365 IC50 = 4900 nM T87675 CMU87F 68239376 IC50 = 13560 nM T87675 CUR2V0 68290592 IC50 > 100000 nM T87675 C7U4VX 68290829 IC50 = 8100 nM T87675 C24IRX 68290838 IC50 > 40000 nM T87675 C2SLT0 68290849 IC50 = 1800 nM T87675 CY60FW 68290875 IC50 > 100000 nM T87675 C7GK8I 68290918 IC50 > 100000 nM T87675 CC8IR2 68290919 IC50 > 100000 nM T87675 CVB70Q 68291007 IC50 = 4200 nM T87675 CN3YX2 68291016 IC50 > 100000 nM T87675 C0OIP9 68291028 IC50 = 21000 nM T87675 C7CZX6 68291099 IC50 > 100000 nM T87675 CEJ26R 68291131 IC50 = 2600 nM T87675 CEZI21 68291184 IC50 > 100000 nM T87675 CY5OU4 68291366 IC50 > 100000 nM T87675 C8CSV6 68291375 IC50 = 28000 nM T87675 C2S0CH 68291448 IC50 > 100000 nM T87675 C8I7GC 68293638 IC50 > 10000 nM T87675 CD56XK 68293660 IC50 > 10000 nM T87675 C2ZLY3 68310278 IC50 = 23000 nM T87675 CY4GV3 68310582 IC50 = 65000 nM T87675 CM5J8Z 68649048 IC50 = 3 nM T87675 CWE54D 68650098 IC50 = 3010 nM T87675 C7GRV2 68755406 IC50 > 10000 nM T87675 C0HA8V 68783839 IC50 = 3 nM T87675 C3GTU1 69762142 IC50 > 10000 nM T87675 CECZ23 70654418 IC50 > 1000 nM T87675 CG50UJ 70654476 IC50 = 330 nM T87675 C4BS5T 70654492 IC50 > 1000 nM T87675 CKP9E6 70654499 IC50 > 1000 nM T87675 CAI3J4 70654537 IC50 = 53 nM T87675 CEXK08 70654539 IC50 > 1000 nM T87675 C5NDK0 70654558 IC50 = 760 nM T87675 C0AP6Q 70654571 IC50 > 1000 nM T87675 CRVS29 70654613 IC50 > 1000 nM T87675 COV46X 70654614 IC50 > 1000 nM T87675 CPF8W3 70654623 IC50 = 160 nM T87675 CVL6N9 70654642 IC50 > 1000 nM T87675 CP0O5A 70654694 IC50 > 1000 nM T87675 C9QS6O 70654709 IC50 > 1000 nM T87675 C4INO3 70654745 IC50 = 940 nM T87675 CC0S3D 70654753 IC50 > 1000 nM T87675 C7F4DB 70654775 IC50 > 1000 nM T87675 C4I8WO 70654805 IC50 = 610 nM T87675 C5LFG2 70654826 IC50 = 500 nM T87675 CA0UR2 70654830 IC50 = 160 nM T87675 CWE94C 70654840 IC50 > 1000 nM T87675 C23AJO 70654866 IC50 > 1000 nM T87675 CS6I4T 70654868 IC50 > 1000 nM T87675 CGU2P6 70654923 IC50 = 1000 nM T87675 C59APG 70654958 IC50 = 430 nM T87675 C2LTI3 70654979 IC50 = 120 nM T87675 C6EK1V 70654997 IC50 = 170 nM T87675 CJAI19 70655010 IC50 > 1000 nM T87675 CX3V5C 70655056 IC50 > 1000 nM T87675 C49KEL 70655062 IC50 = 47 nM T87675 CW8XC7 70655063 IC50 > 1000 nM T87675 CUYK36 70655070 IC50 = 590 nM T87675 CNQ56Y 70657170 IC50 > 1000 nM T87675 C2A4PE 70660513 IC50 = 120 nM T87675 CF92MK 70660523 IC50 = 600 nM T87675 C7QL4R 70660524 IC50 = 320 nM T87675 C5U0EL 70661438 IC50 > 1000 nM T87675 C98FWB 70661441 IC50 = 250 nM T87675 C03CKB 70661448 IC50 = 880 nM T87675 C3NVZ6 70681070 IC50 = 80 nM T87675 C56ZER 70681071 IC50 = 16 nM T87675 CV24XU 70681532 IC50 = 38 nM T87675 CRYW49 70681533 IC50 = 40 nM T87675 CWK7B0 70682875 IC50 > 100000 nM T87675 C1R6HY 70683192 IC50 = 30 nM T87675 CJMQ50 70683427 IC50 <= 4 nM T87675 CDB0H6 70683503 IC50 = 583 nM T87675 C3NCF2 70683641 IC50 = 2 nM T87675 CY51SV 70683642 IC50 = 2 nM T87675 CE86FA 70683706 IC50 = 5520 nM T87675 CD29LB 70684383 IC50 > 12500 nM T87675 C0XPO9 70684384 IC50 = 12500 nM T87675 C6QZ5U 70685271 IC50 = 6 nM T87675 CPTG79 70685272 IC50 = 1.5 nM T87675 C7NP5X 70685550 IC50 = 638 nM T87675 C4PW8O 70685778 IC50 = 11 nM T87675 CN3E5T 70685779 IC50 = 5 nM T87675 C0JU4I 70685852 IC50 = 3040 nM T87675 C6DAJ0 70687420 IC50 = 21 nM T87675 C6FO8B 70687421 IC50 = 10 nM T87675 C9RFK2 70687976 IC50 = 780 nM T87675 CZEN15 70688644 IC50 > 12500 nM T87675 C01WIM 70689476 IC50 = 3 nM T87675 CAE31H 70689940 IC50 = 2 nM T87675 C1IN7G 70689941 IC50 = 2 nM T87675 CXC1H8 70690000 IC50 = 2100 nM T87675 CGA43T 70690710 IC50 = 350 nM T87675 CS1G5L 70691585 IC50 = 17 nM T87675 CDWB98 70691595 IC50 = 40 nM T87675 C5MT8A 70691596 IC50 = 19 nM T87675 CC5A4K 70692098 IC50 = 7.5 nM T87675 CADI76 70692099 IC50 = 20 nM T87675 C16ABH 70692158 IC50 = 650 nM T87675 CW9MY1 70693675 IC50 = 150 nM T87675 C2L6OP 70693678 IC50 = 13 nM T87675 CNRC67 70693679 IC50 = 2 nM T87675 CJZ5E1 70693680 IC50 = 100 nM T87675 C4IV6B 70693993 IC50 <= 4 nM T87675 CY9JR7 70694213 IC50 = 220 nM T87675 CW29QX 70694214 IC50 = 790 nM T87675 C2XV4Q 70694953 IC50 > 100000 nM T87675 C2QJ8X 70695789 IC50 = 25 nM T87675 CPW57H 70695790 IC50 = 87 nM T87675 CC8WG5 70695791 IC50 = 17 nM T87675 C2UMZ0 70695792 IC50 = 17 nM T87675 C1SX4Q 70695793 IC50 = 4 nM T87675 C76JFM 70696269 IC50 = 350 nM T87675 CNI64Y 70696270 IC50 = 2 nM T87675 C03SBG 70696316 IC50 = 3180 nM T87675 CHAY50 70696941 IC50 > 12500 nM T87675 CE1M6V 70702124 IC50 = 24600 nM T87675 CL5T2U 70702125 IC50 = 281 nM T87675 C2YZX3 70702126 IC50 > 50000 nM T87675 CDS8L7 70702127 IC50 = 3.9 nM T87675 C7B2KZ 70702128 IC50 = 19.9 nM T87675 CGF57B 70702129 IC50 = 5.1 nM T87675 C12WBG 70702130 IC50 = 1490 nM T87675 CG1CV9 70702131 IC50 = 3.17 nM T87675 CA9N6S 70702132 IC50 = 376 nM T87675 CK8DC6 70702133 IC50 > 50000 nM T87675 C4YSR1 70702134 IC50 = 1773 nM T87675 CFUY92 70702135 IC50 = 2 nM T87675 CZCP71 70702136 IC50 = 4 nM T87675 CFS53O 70702137 IC50 = 46.6 nM T87675 C3PA9H 70702138 IC50 = 560 nM T87675 CYV57S 70702139 IC50 = 3.3 nM T87675 CY7R5L 70702141 IC50 = 284 nM T87675 C4WHX9 70702142 IC50 = 35 nM T87675 C5RY7I 70702144 IC50 = 30.2 nM T87675 CN4C3L 70702145 IC50 = 8.5 nM T87675 CAH5Z4 70702146 IC50 = 50.2 nM T87675 CVX3W4 70702148 IC50 = 216 nM T87675 CGV53S 70702149 IC50 < 1000 nM T87675 C3CT2W 70702150 IC50 = 1000 nM T87675 CQI41A 70702151 IC50 < 1000 nM T87675 C2T0RP 70702152 IC50 = 71.2 nM T87675 C0Q5XG 70702153 IC50 = 316 nM T87675 CVNR83 70702154 IC50 = 116.5 nM T87675 C4F2HG 70702155 IC50 < 1000 nM T87675 CZ19MK 70702156 IC50 = 253 nM T87675 CR50CX 70702157 IC50 < 1000 nM T87675 CB5Z1F 70702158 IC50 < 1000 nM T87675 CZ19LH 70702159 IC50 < 1000 nM T87675 CL5P4C 70702160 IC50 = 14.4 nM T87675 CXY46F 70702161 IC50 < 1000 nM T87675 CQK2G1 70702162 IC50 = 2.9 nM T87675 CY2P3B 70702164 IC50 = 3 nM T87675 C1IEJ2 70789254 IC50 = 7800 nM T87675 C8T7ZP 70789255 IC50 = 9800 nM T87675 CIQY28 70789751 IC50 = 15 nM T87675 COM14R 71044759 IC50 < 4 nM T87675 CFTP07 71044863 IC50 < 4 nM T87675 CL1HY5 71212233 IC50 = 50000 nM T87675 CKX52R 71212291 IC50 > 100000 nM T87675 C0T2VB 71212317 IC50 = 45000 nM T87675 C5B8NS 71212337 IC50 > 100000 nM T87675 CSN04E 71212395 IC50 > 100000 nM T87675 C1OCW0 71212403 IC50 > 100000 nM T87675 CBX2I4 71212419 IC50 > 100000 nM T87675 CLS4R3 71212434 IC50 > 100000 nM T87675 CTF8M7 71212446 IC50 > 100000 nM T87675 C2Z8CX 71212514 IC50 = 60000 nM T87675 CBT7L3 71212517 IC50 > 100000 nM T87675 C5HB9I 71259491 Ki = 15 nM T87675 C9AF8W 71267243 Ki = 72 nM T87675 CO52YE 71449833 IC50 = 6.6 nM T87675 CB6F8L 71450374 IC50 = 87 nM T87675 CTV95P 71451643 IC50 = 18.7 nM T87675 CIHY26 71452194 IC50 = 9 nM T87675 CHEB80 71452520 IC50 = 13 nM T87675 C3J8BY 71453484 IC50 = 9000 nM T87675 C4FT7D 71454002 IC50 = 130 nM T87675 CLDP69 71454277 IC50 = 40 nM T87675 CCPS09 71454278 IC50 = 93 nM T87675 C47GYB 71454279 IC50 = 30 nM T87675 CTBD38 71454281 IC50 = 45 nM T87675 CK3Y4V 71455743 IC50 = 34 nM T87675 CZT0H5 71455744 IC50 = 26 nM T87675 C1YK3Z 71456034 IC50 = 6 nM T87675 C0FTE7 71456035 IC50 = 22 nM T87675 C2B4HA 71456036 IC50 = 2200 nM T87675 CIUZ98 71456038 IC50 = 35 nM T87675 C7X4MD 71456750 IC50 > 25000 nM T87675 CY8G0F 71459407 IC50 = 4 nM T87675 CBD8Z4 71459408 IC50 = 47 nM T87675 CY8OS1 71459750 IC50 = 27 nM T87675 CP9LF4 71459751 IC50 = 600 nM T87675 C4HOX3 71461167 IC50 = 12 nM T87675 C8CJD0 71461168 IC50 = 54 nM T87675 CXTP95 71461470 IC50 = 564 nM T87675 CMOT45 71461471 IC50 = 45 nM T87675 C27UAH 71462371 IC50 = 4.5 nM T87675 COT2V4 71462903 IC50 = 7 nM T87675 CNI24J 71462904 IC50 = 6 nM T87675 CX1H2S 71462905 IC50 = 11 nM T87675 C7UVZ5 71463198 IC50 = 52 nM T87675 COD87T 71463199 IC50 = 68 nM T87675 CGCT07 71463200 IC50 = 41 nM T87675 CQA4U7 71528975 Ki = 3 nM T87675 CCN01X 71547862 IC50 > 10000 nM T87675 CKF73G 71552560 IC50 = 852 nM T87675 C1NPL0 71552941 IC50 > 30000 nM T87675 CA4PS8 71552942 IC50 > 30000 nM T87675 C3UA9C 71553011 IC50 = 30000 nM T87675 CEZ15Y 71553012 IC50 = 30000 nM T87675 CVIA91 71553085 IC50 = 30000 nM T87675 C1TR3O 71553152 IC50 = 30000 nM T87675 C8MV4P 71554422 IC50 = 66400 nM T87675 CRX81Q 71575642 IC50 > 10000 nM T87675 CHY91V 71578307 IC50 > 100000 nM T87675 C0W2KX 71578373 IC50 > 100000 nM T87675 C6TX9R 71578374 IC50 > 100000 nM T87675 C2D1RN 71578375 IC50 > 100000 nM T87675 C73MEW 71578445 IC50 = 40000 nM T87675 C5NH3V 71578446 IC50 > 100000 nM T87675 CC65WU 71578447 IC50 = 5000 nM T87675 CIP6Q2 71578520 IC50 > 100000 nM T87675 CPJ19D 71578658 IC50 = 60000 nM T87675 C5W0GC 71578744 IC50 > 100000 nM T87675 CLZ59B 71578745 IC50 > 100000 nM T87675 C4A6UT 71614918 IC50 = 471 nM T87675 CCXT12 71614919 IC50 = 88 nM T87675 CB6LS5 71658742 IC50 > 1000 nM T87675 CIN8Q2 71658743 IC50 > 1000 nM T87675 CEY10J 71658863 IC50 = 300 nM T87675 CC40FI 71658864 IC50 = 65 nM T87675 CN7TP5 71659100 IC50 > 1000 nM T87675 C3AMG7 71659101 IC50 > 1000 nM T87675 CD84KP 71659102 IC50 > 1000 nM T87675 CS3Q2M 71659227 IC50 = 98 nM T87675 CYSZ68 71659355 IC50 = 790 nM T87675 CU4C2K 71745477 IC50 = 201 nM T87675 CBW3S7 71745667 IC50 = 18 nM T87675 CG75WF 71745668 IC50 = 124 nM T87675 CI5WR0 71745669 IC50 = 107 nM T87675 CX0WG8 71745670 IC50 = 49 nM T87675 C4ECN6 71745857 IC50 = 49 nM T87675 C91XYQ 71745858 IC50 = 99 nM T87675 C4Q6FE 71815105 IC50 = 551.9 nM T87675 CE04IC 71816173 IC50 = 9 nM T87675 CI8P1V 71816174 IC50 = 270 nM T87675 CWBV20 72164208 IC50 = 6100 nM T87675 CR85FA 72194106 IC50 = 25 nM T87675 C61RNW 72194107 IC50 = 97 nM T87675 CPV6E1 72194108 IC50 = 22 nM T87675 CN8O7C 72194109 IC50 = 34 nM T87675 CMQ9R0 72194110 IC50 = 200 nM T87675 C2BQE0 72194111 IC50 = 147 nM T87675 C85YLK 72194253 IC50 = 10 nM T87675 C0SOK7 72194254 IC50 = 13 nM T87675 C2IT7Z 72194397 IC50 = 12 nM T87675 C2SE6T 72194398 IC50 = 16 nM T87675 C2NFG9 72194399 IC50 = 11 nM T87675 CWD82F 72194400 IC50 = 8 nM T87675 CM8TY6 72194528 IC50 = 112 nM T87675 C5SVI9 72194531 IC50 = 33 nM T87675 CL6PC8 72194532 IC50 = 20 nM T87675 C6JB1F 72194671 IC50 = 7.7 nM T87675 C9V2KY 72196134 IC50 = 32 nM T87675 CMU36W 72196135 IC50 = 46 nM T87675 CM7IS1 72196137 IC50 = 22 nM T87675 C0DL3F 72698602 IC50 < 1 nM T87675 C2XZW3 72708899 IC50 > 40000 nM T87675 CKN46T 72708901 IC50 > 40000 nM T87675 CA6ZB2 72734882 IC50 = 7 nM T87675 CG3E2H 72734883 IC50 = 5 nM T87675 COQC81 72734884 IC50 = 255 nM T87675 C8BW7J 72734885 IC50 = 320 nM T87675 CA58QS 72734886 IC50 = 27 nM T87675 CCP73J 72735062 IC50 = 71 nM T87675 CHJ1P0 72735063 IC50 = 190 nM T87675 CMD43O 72735064 IC50 = 58 nM T87675 CJ4L9T 72735065 IC50 = 204 nM T87675 CID56Z 72735066 IC50 = 45 nM T87675 C5P8ZH 72735248 IC50 = 36 nM T87675 CRMW56 72737416 IC50 = 618 nM T87675 C90PAX 72737417 IC50 = 25840 nM T87675 CFR12B 72737418 IC50 = 211 nM T87675 CRK95J 72737419 IC50 = 1941 nM T87675 C4CT0M 72737420 IC50 = 118 nM T87675 C2T1BW 72737421 IC50 = 743 nM T87675 CQ3O1Z 72737597 IC50 = 4 nM T87675 CA62KV 72737598 IC50 = 5 nM T87675 CG16YE 72771106 IC50 = 600 nM T87675 C3L2WD 73292576 Ki = 480 nM T87675 C0P9LY 73292578 Ki = 180 nM T87675 CJ87SO 73292579 Ki = 2900 nM T87675 CAS80Y 73292746 Ki = 200 nM T87675 C35BCQ 73292749 Ki = 870 nM T87675 C52LFH 73292907 Ki = 54 nM T87675 CZ63BH 73293963 Ki > 5700 nM T87675 C7F0YR 73353451 IC50 = 710 nM T87675 CZN1Y6 73354960 IC50 = 69 nM T87675 CMEV76 74983355 Ki = 460 nM T87675 C47JPV 75202872 IC50 > 50000 nM T87675 C8W2HV 76309526 Ki < 100000 nM T87675 C76NUH 76310311 IC50 > 100000 nM T87675 CP8F0T 76313983 IC50 > 100000 nM T87675 C81ECP 76313984 IC50 = 49000 nM T87675 C7HYN3 76313985 IC50 > 100000 nM T87675 C6D0LO 76316736 Ki < 100000 nM T87675 CRLG27 76317532 IC50 > 100000 nM T87675 CH8Q9D 76324874 IC50 = 72000 nM T87675 CN15WO 76328435 IC50 > 100000 nM T87675 CJ2T9E 76332983 IC50 = 250 nM T87675 C58NAD 76335737 IC50 > 100000 nM T87675 C3HBX9 76335738 IC50 > 50000 nM T87675 CS0CN8 76335739 IC50 > 100000 nM T87675 CPG3A5 86302574 IC50 > 30000 nM T87675 CUNA57 88876306 IC50 = 270 nM T87675 CDW95X 88876318 IC50 = 56 nM T87675 CE6RY9 88876331 IC50 = 150 nM T87675 CT1L6U 88876351 IC50 = 95 nM T87675 C31EBZ 88876355 IC50 = 32 nM T87675 CVEA94 88876366 IC50 = 36 nM T87675 C49LZW 89766055 Ki = 25 nM T87675 C9YWN1 89790691 IC50 = 14 nM T87675 C5Q7UO 90036498 Ki = 780 nM T87675 CC06YJ 90036766 Ki = 520 nM T87675 CO51HL 90037453 Ki = 950 nM T87675 CX4C7W 90037556 Ki = 1700 nM T87675 C28WQY 90431726 IC50 = 16 nM T87675 CY0UC4 90645194 IC50 > 10000 nM T87675 C6WQU2 90645540 Ki = 210 nM T87675 CSD73E 90645541 Ki = 210 nM T87675 C02KJP 90645542 Ki = 290 nM T87675 CE3OV2 90645543 Ki = 2100 nM T87675 CY6L4N 90645544 Ki = 500 nM T87675 C7D5PI 90645545 Ki = 170 nM T87675 C93BGJ 90645546 Ki = 19 nM T87675 C1FSM7 90654763 IC50 = 135 nM T87675 CVH8O1 90654764 IC50 = 113 nM T87675 C7C4EY 90654765 IC50 = 34 nM T87675 CK5R9A 90654766 IC50 = 573 nM T87675 C8P1JL 90654767 IC50 = 228 nM T87675 CYT14Q 90654768 IC50 = 72 nM T87675 C7Q6CY 90654769 IC50 = 101 nM T87675 C7W1JT 90654770 IC50 = 118 nM T87675 CI2M5A 90654771 IC50 = 549 nM T87675 CE62XJ 90654772 IC50 = 5 nM T87675 C12JRV 90654773 IC50 = 127 nM T87675 CP94DI 90666344 IC50 = 13430 nM T87675 CRT7K1 91667406 Ki = 7500 nM T87675 CUCS06 91885526 IC50 <= 100 nM T87675 CACB62 91885527 IC50 <= 100 nM T87675 CRT8F2 92293823 IC50 = 2000 nM T87675 CXS96K 101902488 IC50 = 370 nM T87675 CGB54P 101902999 IC50 = 900 nM T87675 CG62HP 101903000 IC50 = 400 nM T87675 C5N1VZ 102581295 IC50 > 10000 nM T87675 CSD75R 110868446 Ki > 100000 nM T87675 C7ML9C 110868449 Ki > 100000 nM T87675 CICU38 118213763 IC50 = 70 nM T87675 CE49ZI 118475652 IC50 = 43 nM T87675 CS5C8W 118684133 IC50 = 2.1 nM T87675 CY7BI2 118706214 IC50 > 10000 nM T87675 C2IN3C 118710236 IC50 = 203 nM T87675 CE13CO 118710415 IC50 = 1890 nM T87675 CFJ1N6 118710418 IC50 = 690 nM T87675 CF1GH2 118710421 IC50 = 1440 nM T87675 C6O7DN 118710473 IC50 = 720 nM T87675 C6SW3X 118710474 IC50 = 1560 nM T87675 C0D7PO 118710475 IC50 = 1500 nM T87675 CNV92W 118710476 IC50 = 3830 nM T87675 CR7KN3 118710480 IC50 = 1880 nM T87675 CUZL50 118710481 IC50 = 4160 nM T87675 CX0W3J 118710482 IC50 = 1820 nM T87675 C7XE9K 118716988 IC50 = 61 nM T87675 CS8Q2C 118716989 IC50 = 219 nM T87675 C3KLI5 118723185 IC50 > 100000 nM T87675 CG25JP 118725515 IC50 = 11 nM T87675 C6XW9J 118725516 IC50 = 377 nM T87675 CJQE38 118725517 IC50 = 2 nM T87675 CS1FU0 118725519 IC50 = 4 nM T87675 C3QD8O 118725520 IC50 = 4 nM T87675 C6LWF1 118725521 IC50 = 25 nM T87675 CO30HX 118725522 IC50 = 60 nM T87675 CDP96A 118725523 IC50 = 8 nM T87675 CR95GT 118725524 IC50 = 20 nM T87675 C3OP2A 118725526 IC50 = 15 nM T87675 CT8Z0C 118725528 IC50 = 22 nM T87675 CAK4Y3 118725529 IC50 = 21 nM T87675 C46DME 118725530 IC50 = 6 nM T87675 C8I6GM 118725531 IC50 = 11 nM T87675 CG3JU9 118725532 IC50 = 2300 nM T87675 CGB27X 118725533 IC50 = 11 nM T87675 CVTN86 118725534 IC50 = 31 nM T87675 C6ML4Z 118725535 IC50 = 5200 nM T87675 CT7U4L 118734734 IC50 = 12 nM T87675 CYO74T 118734736 IC50 = 43 nM T87675 CQCX41 118737057 IC50 > 10000 nM T87675 CK82IE 121231440 IC50 = 2300 nM T87675 CN81HR 122181799 IC50 > 10000 nM T87675 C2D8UA 122181800 IC50 = 41 nM T87675 CMU6G9 122181801 IC50 = 38 nM T87675 C8DJ3K 122181802 IC50 = 43 nM T87675 CR9FQ7 122181803 IC50 = 320 nM T87675 CTS2C6 122181804 IC50 = 140 nM T87675 CDUA42 122182198 Ki = 17 nM T87675 C30URY 122182199 Ki = 131 nM T87675 CNZG96 122182482 Ki = 893 nM T87675 C9ENM4 122182483 Ki > 5400 nM T87675 CV3X7Z 122182484 Ki > 5400 nM T87675 CV7E8D 122182485 Ki > 5400 nM T87675 CFP8L3 122182486 Ki = 3500 nM T87675 C41VZY 122182487 Ki > 5400 nM T87675 C9Z5AY 122182488 Ki > 5400 nM T87675 CSN1P8 122182489 Ki > 5400 nM T87675 C74VXS 122182490 Ki > 5400 nM T87675 CL3PR1 122182491 Ki > 5400 nM T87675 CFKD32 122191637 IC50 = 493 nM T87675 C5AFZ6 122191639 IC50 = 57 nM T87675 CW5SL7 122191640 IC50 <= 100 nM T87675 CTX98S 122191642 IC50 = 576 nM T87675 CEK1V4 122191643 IC50 = 800 nM T87675 CIR25H 122191977 IC50 <= 100 nM T87675 CFG87R 122191978 IC50 <= 100 nM T87675 C4X7SD 122192466 IC50 > 10000 nM T87675 CJ6RO8 122193596 IC50 > 10000 nM T87675 C18FWG 122197326 IC50 = 468 nM T87675 C8CMZ9 122197327 IC50 = 496 nM T87675 CSP09Z 122197328 IC50 = 82 nM T87675 CYX60U 122197329 IC50 = 157 nM T87675 CE5C3B 122197330 IC50 = 312 nM T87675 C1VGJ2 122197331 IC50 = 436 nM T87675 CBYC49 126617676 IC50 = 192.4 nM T87675 C50QVG 127027240 IC50 = 13700 nM T87675 CHN0C6 127028483 IC50 = 3520 nM T87675 CLQE43 127028484 IC50 = 801 nM T87675 C26ZFL 127028485 IC50 = 2970 nM T87675 CDT31P 127029393 IC50 = 6070 nM T87675 CA4UH3 127029997 IC50 = 5150 nM T87675 C4W7TU 127031218 IC50 = 6430 nM T87675 C0PUM7 127031807 IC50 = 638 nM T87675 CTB34H 127031808 IC50 = 12400 nM T87675 CZ02HG 127031810 IC50 = 15400 nM T87675 CR18NB 127032078 IC50 = 7670 nM T87675 CA6ES3 127053398 IC50 = 284 nM T87675 CRJ04D 127053399 IC50 = 607 nM T87675 CO8Z2N 129900111 EC50 = 38 nM T87675 C0FM1R 130196825 IC50 > 30000 nM T87675 CL26YS 132005219 IC50 = 49 nM T87675 CP32GB 132005220 IC50 = 270 nM T87675 CUN18W 132005225 IC50 = 150 nM T87675 CD84OI 132005228 IC50 = 59 nM T87675 C9VDI0 132005229 IC50 = 23 nM T87675 C7ASP9 132005246 IC50 = 110 nM T87675 C5W9LN 132005323 IC50 = 350 nM T87675 CQ6GO2 132005326 IC50 = 190 nM T87675 CL6E4J 132601725 IC50 = 8300 nM T87675 CF6SG8 134131952 IC50 = 950 nM T87675 CPAW63 134132480 IC50 = 1600 nM T87675 CW94BO 134133208 IC50 = 24 nM T87675 CY0KV9 134134408 IC50 = 1660 nM T87675 CW3NE0 134134901 IC50 = 260 nM T87675 C7HL0T 134135028 IC50 = 6.2 nM T87675 C2K9LG 134135115 IC50 = 25 nM T87675 C8R5MB 134135366 IC50 = 9000 nM T87675 CK5J1Z 134135396 IC50 = 2860 nM T87675 CQ01XS 134135699 IC50 = 15000 nM T87675 CU6QM8 134135714 IC50 > 50000 nM T87675 C0A1MC 134136561 IC50 > 70000 nM T87675 C1MCE8 134136983 IC50 = 480 nM T87675 CIYS07 134137911 IC50 = 6 nM T87675 C2G6CF 134138067 IC50 = 23000 nM T87675 C57JEQ 134138729 IC50 = 52000 nM T87675 CYZ15N 134139678 IC50 = 7800 nM T87675 CI8Y4X 134139821 IC50 = 208 nM T87675 C3F1DI 134140009 IC50 = 3500 nM T87675 CE7Q4G 134140427 IC50 = 1.7 nM T87675 CX5C8B 134140540 IC50 = 66 nM T87675 CJ8S5G 134140875 IC50 = 1290 nM T87675 CFG2B9 134140976 IC50 = 190 nM T87675 CX75IT 134141730 IC50 = 790 nM T87675 C3F1UI 134142262 IC50 = 4 nM T87675 CU4RI0 134142431 IC50 = 220 nM T87675 CN7W4Y 134143295 IC50 = 260 nM T87675 C6YQW8 134143409 IC50 > 200000 nM T87675 C6BZ8J 134143465 IC50 = 12000 nM T87675 C14CDP 134143552 IC50 = 76000 nM T87675 CWB68E 134143937 IC50 = 85 nM T87675 CQJM72 134144731 IC50 = 480 nM T87675 CX3W9U 134145284 IC50 = 480 nM T87675 CX8CE4 134146290 IC50 = 190 nM T87675 C54NEW 134147630 IC50 > 1000 nM T87675 CJ9A1F 134147711 IC50 = 300 nM T87675 CWOX97 134147722 IC50 = 51 nM T87675 CZC9B1 134148432 IC50 = 780 nM T87675 CV3U2O 134148566 IC50 = 380 nM T87675 C7ZUI0 134148651 IC50 = 370 nM T87675 CWQ82I 134148676 IC50 = 314 nM T87675 CN7FJ9 134149620 IC50 = 83 nM T87675 CD62UX 134149816 IC50 = 21000 nM T87675 C6MND7 134149877 IC50 > 1000 nM T87675 C6TE9N 134150616 IC50 = 3300 nM T87675 CFZ7J9 134152243 IC50 = 74 nM T87675 CIP61L 134153498 EC50 = 5.8 nM T87675 C19PLS 134153554 IC50 = 9610 nM T87675 CYF40A 134153592 IC50 = 130 nM T87675 C3XQ6E 134153764 IC50 = 3500 nM T87675 CUT7M5 134153888 IC50 > 200000 nM T87675 CXT13L 134154154 IC50 = 310 nM T87675 C95DNL 134154707 IC50 = 790 nM T87675 CIKC27 134155199 IC50 = 1900 nM T87675 CFN7Q8 134156381 IC50 = 26 nM T87675 CR0PZ9 134156662 IC50 = 600 nM T87675 C8MQ3P 134156839 IC50 = 14000 nM T87675 CZC83Y 134156859 IC50 = 11000 nM T87675 CQ07HK 134157266 IC50 = 60 nM T87675 CT06QO 134157573 IC50 = 4900 nM T87675 CSX26H 134157863 IC50 = 6.2 nM T87675 CGBZ13 134843302 IC50 > 10000 nM T87675 C54FXD 134957362 IC50 > 10000 nM T87675 CLSE63 135398512 IC50 = 58 nM T87675 CS4OW8 135400873 IC50 = 1300 nM T87675 CZ68EL 135414231 IC50 = 16720 nM T87675 CJ65LQ 135423783 IC50 > 100000 nM T87675 C2WL8M 135423784 IC50 > 100000 nM T87675 CNKD13 135423790 IC50 = 2000 nM T87675 C48NWF 135423791 IC50 > 100000 nM T87675 CEVL69 135423792 IC50 = 100000 nM T87675 C6HGC3 135423793 IC50 > 100000 nM T87675 C1W6EI 135423851 IC50 > 100000 nM T87675 CYH51Q 135423852 IC50 > 100000 nM T87675 CYG2V6 135428039 IC50 = 1.5 nM T87675 CK9D4A 135428921 IC50 = 91 nM T87675 CU60YC 135431661 IC50 = 10050 nM T87675 CW5B9U 135432839 IC50 = 5700 nM T87675 C8GZ2B 135449326 Ki > 4000 nM T87675 C4Q5CE 135453643 IC50 < 5000 nM T87675 CUFC14 135502940 IC50 = 69 nM T87675 CTJ48K 135524085 IC50 = 280 nM T87675 CUT1W7 135524168 IC50 = 93 nM T87675 C9ZBY3 135525654 IC50 = 180 nM T87675 CTB7R2 135564980 IC50 = 4 nM T87675 C6QA2T 135566358 IC50 = 10 nM T87675 CJN0Z7 135566360 IC50 = 12 nM T87675 CZY5G2 135566361 IC50 = 5.9 nM T87675 CRJ45X 135589980 IC50 = 8090 nM T87675 C19QOB 135620673 IC50 = 550 nM T87675 C37RUJ 135620674 IC50 = 4200 nM T87675 CD08US 135620675 IC50 > 10000 nM T87675 CADG57 135620676 IC50 > 100000 nM T87675 C4XV9S 135620677 IC50 = 400 nM T87675 CO9L3F 135620678 IC50 > 100000 nM T87675 C0IXJ4 135620680 IC50 = 530 nM T87675 CZ49HM 135723775 IC50 = 590 nM T87675 C6V4DX 135794286 IC50 = 510 nM T87675 CO21NR 135823061 IC50 > 10000 nM T87675 CKU1W0 135834866 IC50 = 430 nM T87675 CV24UR 135873213 IC50 = 1000 nM T87675 CJV08H 135897884 IC50 = 79 nM T87675 C4K3XL 135897887 IC50 = 9.7 nM T87675 C93QJC 135897888 IC50 = 14.9 nM T87675 CX6JV7 135897894 IC50 = 175 nM T87675 C5QUL0 135897897 IC50 = 7.1 nM T87675 CLV7Y8 135897900 IC50 = 41.5 nM T87675 CFJZ14 135897904 IC50 > 10000 nM T87675 CT2UV5 135897905 IC50 = 330 nM T87675 CF0CM3 135909510 IC50 = 70 nM T87675 CVH9A7 135909511 IC50 = 3.5 nM T87675 CWIE69 135909512 IC50 = 2.8 nM T87675 CGSC82 135909513 IC50 = 5.7 nM T87675 CQ1RH0 135909514 IC50 = 13 nM T87675 CX02VW 135909515 IC50 = 26 nM T87675 CE95HA 135922389 IC50 = 300 nM T87675 C3BZ4A 135922390 IC50 > 10000 nM T87675 C8VU0O 135929094 IC50 = 51 nM T87675 CMJ8X5 135929095 IC50 = 110 nM T87675 CF2Z8X 135929096 IC50 = 340 nM T87675 CEP9Y5 135929097 IC50 = 1100 nM T87675 C9N3GW 135929098 IC50 = 870 nM T87675 CVG4I5 135929100 IC50 = 2 nM T87675 C0V2HQ 135929101 IC50 = 72 nM T87675 CIPA79 135937899 IC50 > 10000 nM T87675 C2PAV1 135971426 IC50 = 300 nM T87675 C4RL7Q 135985508 IC50 = 370 nM T87675 CJID74 136013449 IC50 = 15300 nM T87675 CHA4N2 136013680 IC50 > 10 nM T87675 C5XIE8 136026041 IC50 = 33000 nM T87675 CD3U6W 136087130 IC50 = 201.86 nM T87675 C9GMP3 136087133 IC50 = 1400.34 nM T87675 CD1HY8 136087134 IC50 = 328.2 nM T87675 C3UOC4 136087136 IC50 = 1591.65 nM T87675 CG2VJ6 136087137 IC50 > 10000 nM T87675 C7A5SC 136087140 IC50 = 1051.51 nM T87675 C2MDW3 136087152 IC50 > 10000 nM T87675 CI97YR 136087155 IC50 = 495.14 nM T87675 CG05JU 136087156 IC50 = 790.81 nM T87675 CFKB53 136104460 IC50 = 120 nM T87675 C21PTY 136104462 IC50 > 100000 nM T87675 C7XO8B 136104463 IC50 > 100000 nM T87675 C7UH8T 136104464 IC50 > 100000 nM T87675 C7R2PD 136104467 IC50 > 100000 nM T87675 CLEN23 136104468 IC50 > 100000 nM T87675 CWLJ05 136104469 IC50 > 100000 nM T87675 CRI97Z 136126922 IC50 = 68.5 nM T87675 CZUP29 136126923 IC50 = 71.9 nM T87675 CFZ50A 136126924 IC50 = 214.9 nM T87675 C2THI7 136126927 IC50 = 124.9 nM T87675 CG90AI 136126928 IC50 = 91.1 nM T87675 CKU26Y 136126929 IC50 = 321.3 nM T87675 CQ6PT9 136126930 IC50 = 248.8 nM T87675 CQI7M9 136126936 IC50 = 86.1 nM T87675 CWJY91 136126938 IC50 = 28.9 nM T87675 CW4JI1 136126939 IC50 = 45.1 nM T87675 CZ7EX0 136183413 IC50 = 190 nM T87675 CXMG02 136216650 IC50 = 434 nM T87675 CED60I 136216651 IC50 = 147 nM T87675 CPEX14 136216652 IC50 = 118 nM T87675 C1YUD0 136219394 IC50 > 10 nM T87675 C8UH0A 136226786 IC50 = 17.3 nM T87675 C0LO3B 136234657 IC50 = 1134 nM T87675 CU62DL 136234658 IC50 = 77.9 nM T87675 CM63AX 136245248 Ki < 100000 nM T87675 CIU8W3 136254389 IC50 > 10 nM T87675 CFQO70 136375226 IC50 = 700 nM T87675 C3MK9W 136807986 IC50 > 10000 nM T87675 CB6G3P 136966265 IC50 > 10000 nM T87675 CI1E8V 137634241 IC50 = 4050 nM T87675 C6L3HN 137634634 IC50 = 12 nM T87675 C8GQD5 137636872 IC50 = 5300 nM T87675 C8I1KV 137637358 IC50 = 5800 nM T87675 CA8GF2 137637401 IC50 = 210 nM T87675 CZS13Q 137640111 IC50 = 310 nM T87675 C4DRX1 137643187 IC50 = 1050 nM T87675 CBJL60 137643418 IC50 > 10000 nM T87675 CESF45 137644276 IC50 = 430 nM T87675 C3O6XZ 137644537 IC50 > 10000 nM T87675 CGW9I0 137656387 IC50 = 9920 nM T87675 CRH18Z 137656846 IC50 = 293 nM T87675 CM3UF7 137700779 IC50 > 10000 nM T87675 CQR52I 141143841 IC50 = 18 nM T87675 C7GR6C 141483894 IC50 = 188 nM T87675 C0NP3Z 141483896 IC50 = 325 nM T87675 C6VB3O 145925651 IC50 >= 5000 nM T87675 C1RD0T 145949228 IC50 = 90.2 nM T87675 C4RL0N 145949878 IC50 = 21.5 nM T87675 CH9YZ4 145949906 IC50 > 1000 nM T87675 CTH9R6 145950406 IC50 = 17 nM T87675 C4TB3R 145950483 IC50 = 461.9 nM T87675 C95UCZ 145950577 IC50 = 66.3 nM T87675 C2NA5J 145950876 IC50 = 6.3 nM T87675 C07HDJ 145951056 IC50 = 150 nM T87675 C8FPE7 145951250 IC50 = 525 nM T87675 C7ED9I 145952622 IC50 = 233 nM T87675 CHBF06 145952797 IC50 = 52.6 nM T87675 CN2VT9 145953211 IC50 = 7.1 nM T87675 CW3RV1 145953992 IC50 > 10000 nM T87675 CLA54T 145954009 IC50 = 451 nM T87675 CZ7I2Y 145954624 IC50 = 25 nM T87675 C9HUW7 145955353 IC50 = 178 nM T87675 C9VXM4 145955906 IC50 = 55.5 nM T87675 C3IH0W 145956084 IC50 = 232 nM T87675 C8WIA4 145957055 IC50 > 1000 nM T87675 CE90PN 145957225 IC50 = 67 nM T87675 C1JDL3 145957276 IC50 = 198 nM T87675 CUI3W1 145957403 IC50 = 31 nM T87675 CLDG46 145957722 IC50 > 1000 nM T87675 CC10SH 145958079 IC50 = 94 nM T87675 C89XYV 145958579 IC50 = 35 nM T87675 C2W9IL 145959003 IC50 = 23 nM T87675 CV08DO 145959172 IC50 = 9 nM T87675 C70IJE 145959540 IC50 = 67.8 nM T87675 C1U8PV 145959596 IC50 = 247 nM T87675 C7M6XN 145960087 IC50 = 38 nM T87675 C8VPI4 145960125 IC50 = 83.2 nM T87675 CJDG56 145960632 IC50 > 10000 nM T87675 CE21QP 145961382 IC50 > 10000 nM T87675 CI0V8W 145963248 IC50 > 10000 nM T87675 C65YWX 145964882 IC50 = 280 nM T87675 CHC3T0 145965031 IC50 > 10000 nM T87675 CP92ZF 145965329 IC50 = 160 nM T87675 C9HXI4 145966620 IC50 = 1800 nM T87675 CQE9M5 145966810 IC50 = 30 nM T87675 C1EH6C 145967078 IC50 = 560 nM T87675 CK4IV6 145967934 IC50 = 183 nM T87675 CD58LC 145967944 IC50 = 145 nM T87675 CDNC31 145967951 IC50 < 4 nM T87675 C75HDR 145968148 IC50 < 4 nM T87675 C0DEU9 145968159 IC50 < 4 nM T87675 CY7FL8 145968605 IC50 < 4 nM T87675 CRAL38 145968638 IC50 < 4 nM T87675 CRD0G4 145969024 IC50 < 4 nM T87675 CWJ12M 145969155 IC50 = 6 nM T87675 CCH2R0 145969234 IC50 = 118 nM T87675 CL9F4K 145969442 IC50 < 4 nM T87675 C23VZS 145969582 IC50 = 168 nM T87675 CGW5S1 145969844 IC50 = 730 nM T87675 CX70KC 145969955 IC50 < 4 nM T87675 CY43DF 145970132 IC50 < 4 nM T87675 CB8R3A 145970271 IC50 = 610 nM T87675 CIOX52 145970381 IC50 < 4 nM T87675 CQY4I3 145970473 IC50 < 4 nM T87675 CPO34H 145970612 IC50 < 4 nM T87675 C8WX1F 145970663 IC50 < 4 nM T87675 CA03CS 145970720 IC50 < 4 nM T87675 CJ59ZQ 145970874 IC50 = 583 nM T87675 CT73QK 145971147 IC50 < 4 nM T87675 CI9B2A 145971241 IC50 = 228 nM T87675 CUW6I0 145972008 IC50 = 139.3 nM T87675 C40VIL 145972979 IC50 = 660 nM T87675 CQBY19 145974023 IC50 > 10000 nM T87675 C4X7CT 145977420 IC50 = 840 nM T87675 CLA57T 145978300 IC50 = 790 nM T87675 C54FIC 145979195 IC50 = 5 nM T87675 C9DE2V 145979557 IC50 = 191 nM T87675 C8RN4T 145979750 Ki = 30200 nM T87675 CYH41T 145979752 IC50 = 174 nM T87675 CLU75C 145979974 IC50 = 60 nM T87675 CX63VM 145980115 IC50 = 94 nM T87675 C6SM4I 145980334 Ki > 100000 nM T87675 CUA34Y 145980364 IC50 = 69 nM T87675 C05GKB 145980665 IC50 = 132 nM T87675 CNS6I5 145980673 IC50 = 422.9 nM T87675 CR0JD7 145981097 IC50 = 167 nM T87675 CU25SM 145981644 IC50 = 268.5 nM T87675 C7AE4L 145981787 IC50 = 38 nM T87675 C5YCJ0 145982003 IC50 = 46.2 nM T87675 CDB3X6 145982088 IC50 = 34 nM T87675 CQ8A6B 145982177 IC50 = 77.6 nM T87675 CJ8Y9M 145982688 IC50 = 21 nM T87675 CG0B6W 145984157 IC50 = 217 nM T87675 C8C5XL 145984893 IC50 = 9 nM T87675 C9WDL3 145986316 IC50 = 63.1 nM T87675 CE05UV 145986353 IC50 < 4 nM T87675 C64JZF 145986550 IC50 = 72 nM T87675 C8NDE5 145987193 IC50 = 25 nM T87675 C76OKW 145987254 IC50 = 103 nM T87675 C1BR4S 145987787 IC50 = 41 nM T87675 C7LV2F 145987970 IC50 = 108.2 nM T87675 CWYN61 145988204 IC50 = 37 nM T87675 C8XD0B 145988239 IC50 = 101.6 nM T87675 C6S8BD 145988336 IC50 = 827 nM T87675 C61BLV 145988464 IC50 = 744 nM T87675 C93FZG 145988498 Ki = 17300 nM T87675 CSWQ20 145988550 IC50 = 10 nM T87675 C1NS8U 145989128 IC50 = 9 nM T87675 C5EZ1P 145989138 IC50 = 93 nM T87675 C0GNE7 145989369 IC50 = 396.9 nM T87675 CT9D0X 145989541 IC50 = 182.8 nM T87675 CZ6IP8 145989872 Ki > 100000 nM T87675 CI3B9F 145989892 IC50 = 128 nM T87675 CFM97W 145990241 IC50 = 75 nM T87675 C5NB4O 145990292 IC50 = 32 nM T87675 C9T1UF 145990998 IC50 = 24 nM T87675 CQU8G2 145991240 IC50 = 80 nM T87675 CKE21U 145991373 IC50 = 6 nM T87675 CAK5V0 145992869 IC50 = 356.5 nM T87675 CG27SA 145993108 IC50 = 95 nM T87675 C0AHF1 145993112 IC50 = 5951 nM T87675 CE7M4S 145993303 IC50 = 1300 nM T87675 C0YA9U 145993477 IC50 = 192.9 nM T87675 CS3DY6 145993716 IC50 = 70.6 nM T87675 CKT7O3 145993958 Ki = 89600 nM T87675 CJI9H5 155510791 IC50 = 0.8 nM T87675 C2NB1R 155514901 IC50 = 0.14 nM T87675 CJD0Z2 155515276 IC50 = 5.48 nM T87675 C0PG3L 155516058 IC50 = 9.3 nM T87675 C7S4HC 155516408 IC50 = 0.012 nM T87675 C7VB6R 155516420 IC50 = 1.61 nM T87675 CM45EF 155519065 IC50 = 0.59 nM T87675 CEA2C1 155521505 IC50 = 0.18 nM T87675 C1STO9 155525257 IC50 = 0.19 nM T87675 C52FHM 155525581 IC50 = 0.62 nM T87675 CDZ59A 155527907 IC50 = 0.11 nM T87675 CH51PR 155529111 IC50 = 0.012 nM T87675 C90SIO 155535101 IC50 = 0.46 nM T87675 CY2B9K 155538361 IC50 = 0.012 nM T87675 CTSM92 155538441 IC50 = 3 nM T87675 C68GMW 155538446 IC50 > 10000 nM T87675 CT9IM4 155539207 IC50 = 105030 nM T87675 CU2Y4F 155540190 IC50 = 0.438 nM T87675 CM4I2F 155540641 IC50 = 20 nM T87675 CTG40B 155541947 IC50 = 1.86 nM T87675 C9T1YR 155543136 IC50 = 8.5 nM T87675 CC5P1X 155543762 IC50 = 20.1 nM T87675 C27GLF 155545018 IC50 = 2.28 nM T87675 CY6Q8S 155554337 IC50 > 10000 nM T87675 C9XK2G 155559311 IC50 = 0.06 nM T87675 CO2I4P 155559898 IC50 = 22000 nM T87675 D00HVA 11624601 Ki > 6900 nM T87675 D00JMT 210332 IC50 = 110 nM T87675 D00UTU 136104465 IC50 > 100000 nM T87675 D02BXJ 46864270 IC50 > 3000 nM T87675 D03BJB 9549299 IC50 > 10000 nM T87675 D03DZO 11715767 IC50 > 10000 nM T87675 D03YVL 5472558 IC50 > 20000 nM T87675 D04NGS 5330790 IC50 = 11 nM T87675 D04WFN 10202471 IC50 = 67 nM T87675 D04YQF 763936 IC50 = 910 nM T87675 D06AGN 136043837 IC50 = 2300 nM T87675 D06HVH 54613583 IC50 > 10000 nM T87675 D06LJL 9916282 IC50 < 1 nM T87675 D06QWO 14824655 IC50 > 10 ug.mL-1 T87675 D07ADX 54764565 IC50 = 108 nM T87675 D07OXC 11650194 IC50 = 116 nM T87675 D08HFG 24809764 IC50 > 10000 nM T87675 D09HVH 135566652 IC50 > 10 nM T87675 D0A1CM 5281855 IC50 = 2480 nM T87675 D0EU1R 46215815 IC50 = 39810 nM T87675 D0G3SZ 6918469 IC50 = 1.8 ug.mL-1 T87675 D0GN5Z 5281295 IC50 = 850 nM T87675 D0I1IK 136104466 IC50 = 20000 nM T87675 D0J3LR 11634725 Ki = 540 nM T87675 D0ME9B 46868971 IC50 <= 4 nM T87675 D0O6OH 71553154 IC50 = 1550 nM T87675 D0Q3EW 9549303 IC50 = 42 nM T87675 D0Q3NG 11715520 Ki > 6900 nM T87675 D0Q7TO 6419766 IC50 = 28 nM T87675 D0QC0W 9914412 IC50 = 110 nM T87675 D0S7IE 11658882 Ki > 6900 nM T87675 D0T4SJ 10356352 IC50 = 5000 nM T87675 D0T8NU 16757525 IC50 > 4000 nM T87675 D0U8VY 6610278 IC50 = 310 nM T87675 D0UO2H 44556162 IC50 > 10000 nM T87675 D0US9O 45275255 IC50 = 58 nM T87675 D0V6LP 136043836 IC50 = 4300 nM T87675 D0Y0ES 3707 IC50 = 4000 nM T40787 C5EOQ2 446609 Ki = 1 nM T40787 CLW69A 656970 Ki = 0.078 nM T40787 CY63ZA 10126311 Ki = 0.64 nM T40787 C5VPW9 10149815 Ki = 14 nM T40787 CHVJ98 10171596 Ki = 44 nM T40787 C3EC1J 10172355 Ki = 1 nM T40787 C2UJG8 10216038 Ki = 6.4 nM T40787 C4B5VN 10216258 Ki = 90 nM T40787 CF0Q9T 10236743 Ki = 3.2 nM T40787 CG0XB8 10285985 Ki = 720 nM T40787 CS60NW 10287093 Ki = 0.628 nM T40787 C8K7LD 10287147 Ki = 2 nM T40787 C7UT2S 10308245 Ki = 134 nM T40787 CL35CS 23388831 Ki = 1 nM T40787 CG7V9W 24752917 Ki = 5.2 nM T40787 C90ICD 24799124 Ki = 140 nM T40787 C63YXN 24799125 Ki = 2 nM T40787 CX2UG8 24896752 Ki = 368 nM T40787 C0FWP4 24896977 Ki = 130 nM T40787 C8QT3D 24899717 Ki = 10 nM T40787 C4XZO8 24899970 Ki = 12 nM T40787 CV7GD5 44340266 Ki = 0.214 nM T40787 CY0J3P 44398646 Ki = 42 nM T40787 C37TCB 44398647 Ki = 3 nM T40787 C39AUN 44398655 Ki = 0.27 nM T40787 CIC6V9 44398662 Ki = 55 nM T40787 CE4O8G 44398663 Ki = 0.37 nM T40787 C9Y6WA 44398670 Ki = 0.034 nM T40787 CH23BQ 44398697 Ki = 0.16 nM T40787 C6CG9E 44398698 Ki = 8 nM T40787 C83RXS 44398711 Ki = 0.7 nM T40787 CL2X7C 44398714 Ki = 0.01 nM T40787 CK80RJ 44398724 Ki = 0.11 nM T40787 C9WN3O 44398736 Ki = 0.16 nM T40787 C08GMT 44398752 Ki = 0.17 nM T40787 CT76LQ 44398762 Ki = 0.12 nM T40787 C57PKF 44398773 Ki = 0.26 nM T40787 CY13FZ 44398925 Ki > 2000 nM T40787 C6GJA2 44398994 Ki = 0.09 nM T40787 CEA10P 45261513 Ki = 26 nM T40787 CYH26S 45261539 Ki = 0.166 nM T40787 CCZD89 45261550 Ki = 0.266 nM T40787 C41SYP 45264876 Ki = 1 nM T40787 C9PV8G 46937448 Ki = 0.7 nM T40787 CWLN08 46937449 Ki = 0.55 nM T40787 C6H2OI 46939142 Ki = 1.7 nM T40787 C6C3XY 46939144 Ki = 2.1 nM T40787 CO7I0D 46939230 Ki = 2.6 nM T40787 C1MY5I 46939231 Ki = 14 nM T40787 C0M2YK 46939232 Ki = 8 nM T40787 CHC12F 46939233 Ki = 3.2 nM T40787 C64WYO 46939234 Ki = 3 nM T40787 C5T3ON 46939325 Ki = 31 nM T40787 C74CDX 46939328 Ki = 59 nM T40787 CYAL41 46939414 Ki = 71 nM T40787 CIX57L 46939495 Ki = 34 nM T40787 C73GRD 52949329 Ki = 18 nM T40787 CN1W2H 66553590 Ki = 87 nM T40787 CLC9A3 66553591 Ki = 34 nM T40787 CY79UL 66553592 Ki = 602 nM T40787 C7LW1D 66553593 Ki = 34 nM T40787 C5TOR0 66553595 Ki = 105 nM T40787 CNJC63 66553670 Ki = 4.4 nM T40787 C7XM2Y 66553671 Ki = 34 nM T40787 C3GV7O 66553672 Ki = 12 nM T40787 CKA0Y2 66553673 Ki = 87 nM T40787 CFDU56 66553674 Ki = 34 nM T40787 C49AMC 91827502 Ki = 750 nM T27137 D00ENY 33032 Ki = 250 nM T27137 D06LYZ 11559235 IC50 = 10 nM T27137 D0D4OW 57338826 IC50 > 12500 nM T27137 D04JQR 5311261 IC50 = 19000 nM T27137 D0U5CS 213056 EC50 > 100000 nM T27137 D0ZV0R 16660135 IC50 = 5.1 nM T27137 C0MLE4 1217 Ki = 1000000 nM T27137 CL8RX5 1222 Ki = 50000 nM T27137 COM10L 1297 Ki = 30000 nM T27137 CSM0F5 5115 IC50 = 65000 nM T27137 CZBT42 73537 EC50 = 127000 nM T27137 C8NO0Z 77937 EC50 > 1000000 nM T27137 C9H6OS 92136 EC50 > 1000000 nM T27137 CUBH61 101122 EC50 > 1000000 nM T27137 CLMU31 165627 EC50 > 1000000 nM T27137 C34YGT 173564 EC50 > 1000000 nM T27137 CUT07K 177491 Ki = 87000 nM T27137 CR68YU 231345 EC50 > 1000000 nM T27137 C37ROZ 439282 Ki = 150 nM T27137 CO9KU6 443586 Ki = 6600 nM T27137 CPA10R 657896 IC50 = 281 nM T27137 C9DX2A 685051 IC50 = 64000 nM T27137 CGQ2R3 692972 IC50 = 242 nM T27137 C5XE8R 697713 IC50 > 100000 nM T27137 C9P2IQ 699222 IC50 = 20 nM T27137 CIJ7U2 744275 IC50 = 5 nM T27137 C9BC2W 775428 EC50 = 1698.24 nM T27137 CK98RL 1069776 IC50 = 16 nM T27137 C7VCI2 1208332 IC50 = 9.5 nM T27137 CKT3N7 1284324 IC50 = 78 nM T27137 CNI89V 1617110 Ki > 1000000 nM T27137 C0JV7O 2660431 IC50 = 980 nM T27137 C1EP3D 2733518 Ki = 329000 nM T27137 C5F8YH 2733519 EC50 = 210000 nM T27137 C1B8WE 2862916 EC50 = 4786.3 nM T27137 CZV0P5 3246152 Ki = 10000 nM T27137 CP5C1A 3931705 Ki = 8800 nM T27137 CGWD04 4125492 EC50 = 1400 nM T27137 C29ANP 4166844 EC50 > 10000 nM T27137 COJV81 4521898 EC50 > 10000 nM T27137 CZ1Q5P 4694355 Ki > 1000000 nM T27137 CWK7X4 4694356 Ki = 860000 nM T27137 C05WNA 5310956 Ki = 50000 nM T27137 CGMN04 5311262 Ki = 350 nM T27137 CL5IB3 5311460 IC50 = 40000 nM T27137 CZ3G8M 6603702 IC50 = 214000 nM T27137 CW4HF2 6603885 EC50 = 6000 nM T27137 C7J6KQ 6604704 EC50 > 300000 nM T27137 C9INH1 6604707 EC50 > 1000000 nM T27137 CD68LI 6604795 Ki > 1000000 nM T27137 C6QSA9 7157252 Ki > 270000 nM T27137 CIA9B5 9794218 IC50 > 100000 nM T27137 C5WAT4 9815955 Ki = 6000 nM T27137 CL8JI1 9837114 EC50 > 1000000 nM T27137 C8NWE5 9844204 Ki = 5700 nM T27137 CH54PF 9991661 Ki = 135000 nM T27137 C0GN6F 10012356 Ki = 250000 nM T27137 CQJP31 10012681 Ki > 1000000 nM T27137 CUN9V7 10036599 IC50 = 73000 nM T27137 CAU7N4 10059959 Ki > 270000 nM T27137 CZ71GJ 10085578 IC50 = 51 nM T27137 C8H3UO 10176324 EC50 > 100000 nM T27137 C9XQK6 10198133 EC50 > 100000 nM T27137 CL4NP9 10198359 IC50 = 76000 nM T27137 CAZ8P0 10198574 Ki > 270000 nM T27137 CFDX64 10241509 EC50 > 300000 nM T27137 CBCE85 10245890 IC50 = 20 nM T27137 CZ7A5Y 10263168 Ki = 110000 nM T27137 CX12HM 10330132 Ki > 1000000 nM T27137 CZ09YG 10358265 IC50 > 300000 nM T27137 CQ1L0O 10359073 Ki > 300000 nM T27137 C8FU6G 10442268 EC50 = 257000 nM T27137 CYL91R 10456810 IC50 > 100000 nM T27137 C3KHU7 10465017 EC50 > 1000000 nM T27137 CK9MN4 10465478 EC50 > 1000000 nM T27137 CO9MK3 10489913 Ki = 60000 nM T27137 C34LSX 10489914 Ki > 270000 nM T27137 CU9BA6 10513894 Ki = 44000 nM T27137 CQGZ24 10513895 Ki > 270000 nM T27137 CYC9W8 10513896 Ki > 270000 nM T27137 CH9VN3 10560963 EC50 = 232000 nM T27137 CDN69Z 10609381 EC50 > 1000000 nM T27137 C57GCR 10656383 Ki > 1000000 nM T27137 C8FP7I 10681240 Ki > 270000 nM T27137 CC6T7Z 10704895 Ki > 270000 nM T27137 CC7JP9 10704896 Ki > 270000 nM T27137 CC2PB0 10752213 Ki = 260000 nM T27137 C27KWL 10752214 Ki = 205000 nM T27137 CQTF38 10775369 EC50 = 121000 nM T27137 C9BK1A 10846649 EC50 = 1600 nM T27137 CU1M0Y 10851012 IC50 = 300 nM T27137 C71RET 11174504 IC50 = 9 nM T27137 CKDH04 11177701 IC50 = 62 nM T27137 C1AZ6P 11185961 IC50 = 74 nM T27137 C2HTB4 11186076 IC50 = 85 nM T27137 CU63ER 11209923 IC50 = 18 nM T27137 CB03EC 11220954 IC50 = 16 nM T27137 CS20IL 11232604 IC50 = 6 nM T27137 C0DK4N 11232687 IC50 = 2 nM T27137 CBRM85 11232871 IC50 = 7 nM T27137 CAN85Y 11255377 IC50 = 3 nM T27137 C0T4SF 11256015 IC50 = 4 nM T27137 CKJ70T 11313361 Ki = 0.34 nM T27137 C8F4QH 11324832 IC50 = 85 nM T27137 CUV4Z0 11325594 IC50 = 5.5 nM T27137 CQ78GX 11347669 IC50 = 160 nM T27137 CL7A2C 11347844 IC50 = 174 nM T27137 CJ4V0I 11382171 IC50 = 450 nM T27137 CAP47E 11383509 IC50 = 6310 nM T27137 CYTN81 11403753 IC50 = 80 nM T27137 CC51BG 11414108 IC50 > 10000 nM T27137 CVFJ08 11450605 IC50 = 29 nM T27137 CBO63D 11461116 IC50 = 1 nM T27137 CK2F5L 11474450 IC50 = 191 nM T27137 CM0GP3 11483517 IC50 > 10000 nM T27137 CR91LD 11483690 IC50 = 0.56 nM T27137 C98DXE 11485531 IC50 = 105 nM T27137 C90BXG 11493585 IC50 = 82 nM T27137 CWQU24 11493897 IC50 = 140 nM T27137 CTB4K0 11501188 IC50 = 251 nM T27137 CI6G2R 11501465 IC50 = 44 nM T27137 C60PZU 11515679 IC50 = 130 nM T27137 CY8SI0 11515957 IC50 = 13 nM T27137 CQNE82 11530673 IC50 = 180 nM T27137 CY90XO 11530971 IC50 = 84 nM T27137 C9FGB7 11537767 IC50 = 167 nM T27137 C5TG6U 11537814 IC50 = 122 nM T27137 CQ5H1B 11543205 EC50 > 1000000 nM T27137 CSFO10 11552320 IC50 = 407 nM T27137 CZVQ09 11560185 IC50 = 32 nM T27137 CV7FE9 11565466 IC50 = 632 nM T27137 CE2P8Y 11566478 IC50 = 183 nM T27137 C6XH5Z 11574901 IC50 = 4 nM T27137 C23SQX 11581985 IC50 = 71 nM T27137 CTBF56 11582178 IC50 = 99 nM T27137 CW8M5V 11588590 IC50 = 87 nM T27137 C5Z9KA 11594849 IC50 = 335 nM T27137 CGX8F6 11596869 EC50 > 12500 nM T27137 C3J6UO 11609353 IC50 = 5 nM T27137 CMBS38 11631279 IC50 = 26 nM T27137 C9F3WR 11639176 IC50 = 37 nM T27137 CCET62 11639210 IC50 = 306 nM T27137 CD5Q9A 11652895 IC50 = 1460 nM T27137 CVYR03 11654379 IC50 = 101 nM T27137 CU58GV 11660511 IC50 = 49 nM T27137 C1P3XR 11660540 IC50 = 41 nM T27137 C0MOJ5 11661106 IC50 = 45 nM T27137 CJ85FI 11666576 IC50 = 167 nM T27137 CGR90L 11667270 IC50 = 23 nM T27137 CO3X5A 11674352 IC50 = 39 nM T27137 C6ZB8C 11681575 IC50 = 98 nM T27137 C0VRM1 11681680 IC50 = 482 nM T27137 C65FWA 11681681 IC50 = 139 nM T27137 CTAP95 11682046 IC50 = 113 nM T27137 CLVO83 11682866 IC50 > 100000 nM T27137 CJCZ59 11688880 IC50 = 17 nM T27137 C97SMI 11695588 IC50 = 50 nM T27137 C1ILY6 11695769 IC50 = 50 nM T27137 CF6LG4 11695894 IC50 = 7.2 nM T27137 CR5B3L 11696595 IC50 = 76 nM T27137 CND69H 11702918 IC50 = 19 nM T27137 C5HFM9 11703031 IC50 = 949 nM T27137 CX8O6F 11716890 IC50 = 16 nM T27137 CS0A4X 11717278 IC50 = 9 nM T27137 CY2VL6 11717319 IC50 = 39 nM T27137 CASI54 11768848 EC50 > 1000000 nM T27137 CP7QF3 11772069 IC50 = 3.3 nM T27137 C96YUT 11820180 Ki = 184000 nM T27137 CJ4WL9 15207262 IC50 = 2400 nM T27137 CSW38G 15420544 EC50 > 10000 nM T27137 CV26IE 15953801 IC50 = 0.8 nM T27137 CPC09T 15985249 IC50 = 3.6 nM T27137 CLY8U2 16038338 IC50 = 10 nM T27137 CW6M4V 16038352 IC50 = 16.8 nM T27137 CPQE54 16117042 IC50 = 55 nM T27137 CSUW31 16117046 IC50 = 27 nM T27137 CDY9Z0 16117168 IC50 = 68 nM T27137 CF3C1I 16117172 IC50 = 47 nM T27137 C3YTO0 16117300 IC50 = 75 nM T27137 C7DNZ1 16117303 IC50 = 88 nM T27137 C2LTK8 16117432 IC50 = 34 nM T27137 C8CNU5 16117433 IC50 = 88 nM T27137 C3U0VK 16117434 IC50 = 31 nM T27137 CJEN28 16117979 IC50 = 8.1 nM T27137 C64FAY 16118120 IC50 = 4.7 nM T27137 CSLK82 16118121 IC50 = 5 nM T27137 C3WI2G 16118122 IC50 = 8.2 nM T27137 C6X3ED 16118123 IC50 = 5.7 nM T27137 C4R1BK 16118124 IC50 = 3.1 nM T27137 CFU1R8 16118126 IC50 = 6.3 nM T27137 C48IBM 16118256 IC50 = 5.4 nM T27137 CA8DR6 16118397 IC50 = 4.4 nM T27137 C6X5HW 16118398 IC50 = 3 nM T27137 C9MED6 16118400 IC50 = 9.8 nM T27137 CKO84B 16118535 IC50 = 7.7 nM T27137 CC6U5Y 16118536 IC50 = 15 nM T27137 C8OG2C 16118539 IC50 = 17 nM T27137 C06BVY 16118540 IC50 = 2 nM T27137 C52XAF 16118542 IC50 = 3.4 nM T27137 C4X6EZ 16118680 IC50 = 0.4 nM T27137 CE0VB6 16118681 IC50 = 5.2 nM T27137 CY4I3R 16118682 IC50 = 3.9 nM T27137 C62FQV 16118685 IC50 = 2 nM T27137 CKHQ02 16118686 IC50 = 2.3 nM T27137 CZ1Y2D 16118812 IC50 = 10 nM T27137 C87ZLF 16118813 IC50 = 14 nM T27137 CKG3B4 16118815 IC50 = 6.4 nM T27137 CPRT86 16118816 IC50 = 15 nM T27137 C7R1BP 16118817 IC50 = 12 nM T27137 C7FX9R 16118818 IC50 = 6.7 nM T27137 C6DJG9 16118942 IC50 = 15 nM T27137 CS7BC5 16118943 IC50 = 35 nM T27137 C6KDF7 16118945 IC50 = 54 nM T27137 CX54MZ 16118946 IC50 = 79 nM T27137 C9UOD4 16118949 IC50 = 85 nM T27137 C2K3UY 16659642 IC50 = 37.6 nM T27137 CN5C2Q 16659643 IC50 = 0.4 nM T27137 C0M8NP 16659645 IC50 = 0.7 nM T27137 C7RHT2 16659646 IC50 = 4.9 nM T27137 CAH3Y2 16659647 IC50 = 541 nM T27137 C4KJ8T 16659798 IC50 = 636 nM T27137 CIJ3A0 16659799 IC50 = 446 nM T27137 C8ZXU6 16659804 IC50 = 24.4 nM T27137 C71WGT 16659805 IC50 = 12 nM T27137 CB17RP 16659963 IC50 = 6 nM T27137 C1NL8Q 16659964 IC50 = 9.8 nM T27137 CWT36L 16659966 IC50 = 2.2 nM T27137 C8IX9D 16659968 IC50 = 5.3 nM T27137 C80LVT 16660140 IC50 = 3.7 nM T27137 CZ2IS9 16660294 IC50 = 1.8 nM T27137 CI86GL 16660467 IC50 = 2.4 nM T27137 CM5NP1 16661404 IC50 = 62 nM T27137 C8GER0 16661405 IC50 = 83 nM T27137 CQDW57 16661406 IC50 = 80 nM T27137 C1IJK8 16661408 IC50 = 6 nM T27137 C6UAE0 16661409 IC50 = 49 nM T27137 CIX6M5 16661726 IC50 = 49 nM T27137 CW5BG1 16661728 IC50 = 18 nM T27137 CV5EA3 16661729 IC50 = 81 nM T27137 CK1X2Y 16730193 IC50 = 5 nM T27137 C7PS0F 17228330 IC50 > 100000 nM T27137 C04GUC 17758443 Ki = 34000 nM T27137 C0Z2XO 17758444 Ki = 254000 nM T27137 CGZF13 17758445 Ki > 300000 nM T27137 C1GSZ4 17758449 Ki > 300000 nM T27137 CZW76I 17758450 Ki > 300000 nM T27137 CT64UF 17758554 Ki = 77000 nM T27137 C3X6WB 17758555 Ki > 300000 nM T27137 C1AD2J 17758556 Ki > 300000 nM T27137 CS5B7A 18138918 IC50 = 630 nM T27137 C6FTH4 19705292 IC50 = 9.8 nM T27137 CD6PM1 22268047 IC50 = 25000 nM T27137 CBV62I 22708855 EC50 = 9300 nM T27137 C0K9DR 22884216 IC50 = 57000 nM T27137 CTQ5X8 23634169 IC50 = 1.5 nM T27137 CJ3ZL8 23634170 IC50 = 1 nM T27137 CYKF96 23634174 IC50 = 1 nM T27137 CW2PD7 23634249 IC50 = 1.8 nM T27137 CKL4B6 23634254 IC50 = 1.1 nM T27137 C5E1DJ 23634325 IC50 = 1.9 nM T27137 CX3BC2 23634326 IC50 = 2 nM T27137 CZ4EC2 23655076 IC50 = 127 nM T27137 CJ18UB 23657393 IC50 = 2.4 nM T27137 CBF6J9 24815439 EC50 > 15848.93 nM T27137 C0XQA3 24884476 IC50 = 9 nM T27137 CDXH35 24967422 EC50 = 316.23 nM T27137 CA3D2O 24967783 EC50 = 794.33 nM T27137 CWV80G 25067015 Ki = 110 nM T27137 CNF72Q 44190035 IC50 > 10000 nM T27137 C3WL6N 44230992 IC50 = 279 nM T27137 CLJN80 44237734 EC50 = 1000 nM T27137 C09VPJ 44243470 IC50 = 644 nM T27137 CL13FV 44302605 IC50 > 300000 nM T27137 C03QML 44302608 IC50 > 300000 nM T27137 C2H6QV 44302609 IC50 = 133000 nM T27137 CP1QS5 44302686 IC50 = 238500 nM T27137 CR0JD5 44302687 IC50 > 300000 nM T27137 C0V9DN 44302818 IC50 > 300000 nM T27137 CDM1P2 44302819 IC50 > 300000 nM T27137 C1GV9Q 44302837 IC50 > 300000 nM T27137 C1FJU0 44302855 IC50 > 300000 nM T27137 C34AVQ 44302856 IC50 > 300000 nM T27137 CLF56U 44302896 IC50 > 300000 nM T27137 C9Y6QA 44302913 IC50 > 300000 nM T27137 CC7BN3 44302929 IC50 > 300000 nM T27137 CKL1M8 44302930 IC50 > 300000 nM T27137 C9U0NH 44302931 IC50 > 300000 nM T27137 CD5XY2 44302932 IC50 > 300000 nM T27137 C5ROF1 44322518 Ki = 750000 nM T27137 CFTA38 44322537 Ki > 100000 nM T27137 C7E8SH 44322745 Ki = 500000 nM T27137 CWV7F0 44322840 Ki > 100000 nM T27137 CGL0Z3 44322843 Ki > 1000000 nM T27137 C2SKJ1 44322921 Ki = 1600 nM T27137 CR1OL6 44328753 IC50 = 57000 nM T27137 CUA80G 44328850 IC50 > 100000 nM T27137 C2SH0O 44329024 IC50 > 100000 nM T27137 CX0Y4F 44329029 IC50 = 5700 nM T27137 C76LOU 44329031 IC50 = 54900 nM T27137 CCV4N5 44329032 IC50 = 18000 nM T27137 CDP86T 44329033 IC50 > 100000 nM T27137 C9V5XC 44329042 IC50 > 100000 nM T27137 CHV03D 44338561 EC50 > 1000000 nM T27137 CV9K5Y 44387697 IC50 = 8 nM T27137 C7H8RT 44387705 IC50 = 5000 nM T27137 CP2QD8 44387711 IC50 > 10000 nM T27137 CTH37F 44387723 IC50 = 1175 nM T27137 CA9VD1 44416124 IC50 >= 10000 nM T27137 C36JLH 44421618 IC50 = 8500 nM T27137 C8C7GX 44430062 IC50 = 3.981 nM T27137 CS42AM 44430063 IC50 = 31.62 nM T27137 CK56QZ 44430064 IC50 = 19.95 nM T27137 C7EI5M 44430065 IC50 = 199.53 nM T27137 C6T5NE 44430066 IC50 = 158.49 nM T27137 C4F5UX 44430067 IC50 = 100 nM T27137 CVXB82 44430068 IC50 = 1000 nM T27137 CF2ED8 44430069 IC50 = 316.23 nM T27137 CVT6Y7 44430070 IC50 < 10000 nM T27137 C27JQH 44435349 IC50 = 5.9 nM T27137 CN8RC6 44442420 IC50 > 100000 nM T27137 CJD2R3 44442421 IC50 > 100000 nM T27137 CS6HF7 44442422 IC50 = 800 nM T27137 CVXY04 44442423 IC50 = 760 nM T27137 CE36NS 44442424 IC50 = 91 nM T27137 CPXN04 44442425 IC50 = 240 nM T27137 C0B5VU 44442426 IC50 = 520 nM T27137 CKRV87 44442427 IC50 > 100000 nM T27137 CH4C8M 44442428 IC50 = 350 nM T27137 CL4J2I 44442429 IC50 = 180 nM T27137 C5FIC0 44442430 IC50 = 220 nM T27137 CQ74SX 44442432 IC50 = 1100 nM T27137 C5F9EB 44442433 IC50 > 100000 nM T27137 C34NJZ 44442434 IC50 = 230 nM T27137 CBEQ37 44442435 IC50 = 9800 nM T27137 CJ39IF 44442436 IC50 > 100000 nM T27137 C3CE4J 44447970 IC50 = 1000 nM T27137 C32FHY 44447971 IC50 = 6 nM T27137 CZG3T6 44569826 Ki > 1000000 nM T27137 CJ28TF 44569827 Ki = 210000 nM T27137 CFZ64A 44569859 Ki = 59000 nM T27137 CUW74T 44569860 Ki > 1000000 nM T27137 C2IKO1 44569861 Ki > 300000 nM T27137 CADV97 44569862 Ki > 1000000 nM T27137 C0DJ2Z 44588385 IC50 = 6.3 nM T27137 CQ9IK3 44588386 IC50 = 18 nM T27137 C8QXF5 44588425 IC50 = 16 nM T27137 C2ZS9A 44588426 IC50 = 11 nM T27137 C58NLO 44588427 IC50 = 590 nM T27137 CMEC89 44588428 IC50 = 57 nM T27137 C1SBZ0 44588429 IC50 = 120 nM T27137 CVKW41 44588460 IC50 = 49 nM T27137 CTJA65 44588461 IC50 = 55 nM T27137 CL24ZS 44588462 IC50 = 220 nM T27137 CP5O4L 44588463 IC50 = 2.6 nM T27137 CKTI06 44588464 IC50 = 7 nM T27137 CFAM64 45082292 EC50 = 6100 nM T27137 C2Y4NF 45484850 IC50 = 1500 nM T27137 CH2YV1 45484871 IC50 = 33 nM T27137 C4VPA7 45484872 IC50 = 2400 nM T27137 CAM93W 45484880 IC50 = 210 nM T27137 CVP16D 45484889 IC50 = 470 nM T27137 CR3J5H 45484897 IC50 = 170 nM T27137 C0H8JT 45484905 IC50 = 880 nM T27137 C8ZK6I 45484911 IC50 = 1800 nM T27137 C7W8RH 45484920 IC50 = 22 nM T27137 C91MAT 45484921 IC50 = 69 nM T27137 COB15H 45484928 IC50 = 3900 nM T27137 CA69XL 45484929 IC50 = 11 nM T27137 COX0G6 45484935 IC50 = 2.6 nM T27137 CANT85 45484964 IC50 = 250 nM T27137 C8WV6H 45484965 IC50 = 4.9 nM T27137 CT6Q9E 45484973 IC50 = 300 nM T27137 CLDS91 45486747 IC50 = 100 nM T27137 CD19ZV 45486748 IC50 = 130 nM T27137 CYSU62 45486754 IC50 > 10000 nM T27137 CZVR14 45486755 IC50 = 230 nM T27137 C7IV3E 45486758 IC50 = 2000 nM T27137 CZP87H 45486764 IC50 = 210 nM T27137 CI6NA2 45486778 IC50 = 77 nM T27137 CZL5F9 45486781 IC50 = 1500 nM T27137 CMD32J 45486799 IC50 > 10000 nM T27137 C0N2HC 45486816 IC50 = 1500 nM T27137 C10VGE 45486817 IC50 = 5700 nM T27137 C31PAF 46700737 EC50 > 10000 nM T27137 CGS4F2 46836713 EC50 > 10000 nM T27137 CIGD23 46870038 EC50 = 316.23 nM T27137 CY5Q8L 46886118 IC50 > 1000 nM T27137 C1B5XO 46886119 IC50 > 1000 nM T27137 C4YD2C 46886120 IC50 = 326 nM T27137 CM9KV2 46886135 IC50 = 16 nM T27137 CR1O4K 46886136 IC50 = 188 nM T27137 CYO8Z9 46886137 IC50 = 68 nM T27137 CJ57LM 46886138 IC50 = 11 nM T27137 CAF9X1 46886139 IC50 > 1000 nM T27137 CG6W8P 46886140 IC50 = 3.1 nM T27137 C6SYU4 46886169 IC50 > 1000 nM T27137 CJM4V9 46927956 EC50 > 100000 nM T27137 C9SD8H 46947824 EC50 = 251.19 nM T27137 CP8E4O 49788655 IC50 = 11 nM T27137 CMI0J4 49788727 IC50 = 21 nM T27137 CU8O9W 49788729 IC50 = 87 nM T27137 C9QH1W 49788731 IC50 = 41 nM T27137 C2EB4M 49788806 IC50 = 105 nM T27137 CV6F9U 49799828 IC50 > 300000 nM T27137 CR65GE 49800187 EC50 = 125.89 nM T27137 CWE2O4 51033723 IC50 > 10000 nM T27137 CE4KP1 51050257 Ki > 10000 nM T27137 CN9RK5 51116040 EC50 = 549.54 nM T27137 CRG53A 52203651 EC50 = 97 nM T27137 CORM67 52941383 EC50 = 1584.89 nM T27137 CHCO75 52941496 EC50 = 794.33 nM T27137 CU2WT8 52941697 IC50 = 32 nM T27137 CBS8J3 52942778 EC50 = 3162.28 nM T27137 C1RE3W 52942855 EC50 = 1000 nM T27137 C3MD2Y 52943768 EC50 = 794.33 nM T27137 CN07TX 52944782 EC50 > 100000 nM T27137 CPWF70 52945134 EC50 = 251.19 nM T27137 C6LQU4 52945583 EC50 = 1584.89 nM T27137 C45IUO 52946206 EC50 = 1584.89 nM T27137 CDES08 52946415 EC50 = 630.96 nM T27137 CO3GF6 52947461 EC50 = 1584.89 nM T27137 C2FZH4 52947627 EC50 = 501.19 nM T27137 C0E4GW 52947637 EC50 = 1584.89 nM T27137 C5O8SR 52948725 EC50 = 2511.89 nM T27137 C7DM1B 52949785 EC50 = 630.96 nM T27137 C4YW5J 52949928 EC50 = 1995.26 nM T27137 CN1HU8 53235518 EC50 > 10000 nM T27137 CY58NO 53240406 EC50 > 25000 nM T27137 C5KAM7 53316848 Ki = 2 nM T27137 CW36CH 53322382 EC50 > 10000 nM T27137 CZ03BQ 54579958 IC50 = 7.7 nM T27137 CVM2Z7 54579959 IC50 = 219 nM T27137 COLN14 54580485 IC50 = 12.6 nM T27137 C5O1LV 54580945 IC50 = 955 nM T27137 CHFO58 54580946 IC50 = 53 nM T27137 C3ST8U 54580947 IC50 = 33 nM T27137 C1VR9A 54580948 IC50 = 13 nM T27137 CDY0N6 54580949 IC50 = 314 nM T27137 CE3VP1 54581505 IC50 = 6.9 nM T27137 CIHC67 54582001 IC50 > 30000 nM T27137 CCR0O3 54582002 IC50 = 12.4 nM T27137 C2V1FR 54582003 IC50 = 4.6 nM T27137 CSF8T1 54582004 IC50 = 3.9 nM T27137 C0O6PC 54582005 IC50 = 85 nM T27137 CYN49G 54582006 IC50 = 137 nM T27137 CQ73VM 54582007 IC50 = 358 nM T27137 CY9XF3 54582494 IC50 = 103 nM T27137 CM6QA5 54582942 IC50 = 9.6 nM T27137 C19GTC 54582943 IC50 = 10.7 nM T27137 CCY49K 54582944 IC50 = 17 nM T27137 CWMT03 54582945 IC50 = 8.2 nM T27137 CZ17AI 54582946 IC50 = 209 nM T27137 CX4CA2 54582947 IC50 = 171 nM T27137 CPZ83T 54583474 IC50 = 43 nM T27137 COAT86 54583942 IC50 = 106 nM T27137 CTG4X9 54583943 IC50 = 21 nM T27137 CZ5K2Y 54584442 IC50 = 11 nM T27137 CXP59T 54584443 IC50 = 6.8 nM T27137 C23PDM 54584887 IC50 = 10.8 nM T27137 C8PW4R 54584888 IC50 = 14.5 nM T27137 CY3P6J 54584889 IC50 = 72 nM T27137 CB5MH3 54584890 IC50 = 8.9 nM T27137 CSBE97 54584891 IC50 = 3 nM T27137 CD26YU 54584892 IC50 = 45 nM T27137 C6D9YF 54585403 IC50 = 4.4 nM T27137 C5CBA9 54585404 IC50 = 10.6 nM T27137 CR5K0W 54585405 IC50 = 16.4 nM T27137 CB5Z9Y 54585406 IC50 = 10.4 nM T27137 C8AJ3Y 54585457 Ki = 4.8 nM T27137 CS1X5M 54585850 IC50 = 12.5 nM T27137 C93WBA 54585851 IC50 = 6.8 nM T27137 CFM8Q2 54585852 IC50 = 212 nM T27137 C6WK1O 54586361 IC50 = 60 nM T27137 CHU13F 54586362 IC50 = 66 nM T27137 CE3X5Z 54586363 IC50 = 241 nM T27137 CF94LX 54586817 IC50 = 3.8 nM T27137 CLPR07 54586818 IC50 = 16 nM T27137 CILU43 54587386 IC50 = 196 nM T27137 C73SDV 55726220 EC50 < 10000 nM T27137 C0T6OW 55778597 EC50 > 10000 nM T27137 CY70XE 57391670 IC50 = 203 nM T27137 C48ZCK 57397023 IC50 = 118 nM T27137 CW56RI 57398691 IC50 > 1000 nM T27137 C0RPC1 57398788 IC50 > 1000 nM T27137 C3CBY4 57400362 IC50 = 133 nM T27137 CBO04Q 57402169 IC50 > 1000 nM T27137 C53VOY 57403924 IC50 = 124 nM T27137 C3NMU1 57403925 IC50 = 192 nM T27137 CWK1D4 57404255 IC50 = 9 nM T27137 CC8N9R 57559280 IC50 = 3 nM T27137 CLUD90 57559287 IC50 = 1 nM T27137 CZ6IE0 57559301 IC50 = 8 nM T27137 CL0R2Q 57559313 IC50 = 2 nM T27137 CFBX49 57559370 IC50 = 86 nM T27137 CVN1K2 57559437 IC50 = 7 nM T27137 C0KGQ3 57559476 IC50 = 16 nM T27137 CWTH50 57559504 IC50 = 20 nM T27137 CLP93Z 57559545 IC50 = 4 nM T27137 CC69EG 57559552 IC50 = 204 nM T27137 CZWP49 57559572 IC50 = 9 nM T27137 C6OS5V 57559578 IC50 = 24 nM T27137 CNBR74 57559597 IC50 = 5 nM T27137 C4Z7LT 57559648 IC50 = 14 nM T27137 C7ORF4 57881625 IC50 = 3 nM T27137 CTY0F2 57881665 IC50 = 7 nM T27137 CL6M7D 57881666 IC50 > 1000 nM T27137 CDF1Y3 57881696 IC50 > 1000 nM T27137 CF8VP5 57881707 IC50 = 12 nM T27137 C2AY8B 57881727 IC50 = 9 nM T27137 CU28WN 57881747 IC50 > 1000 nM T27137 C7Y6JI 57881754 IC50 = 5 nM T27137 C1CT0P 57881755 IC50 > 1000 nM T27137 C9APU5 57881773 IC50 = 30 nM T27137 C7HNR6 57881781 IC50 > 1000 nM T27137 C0F2YG 57881805 IC50 > 1000 nM T27137 CYRM53 57881818 IC50 = 19 nM T27137 CW48BK 57881822 IC50 = 154 nM T27137 C8AJR6 57881832 IC50 = 70 nM T27137 CZ4XS9 57881851 IC50 = 192 nM T27137 C2Z9KP 57881896 IC50 = 277 nM T27137 CNIW19 57881906 IC50 = 82 nM T27137 CUKR86 57881945 IC50 = 15 nM T27137 CQCI36 57881958 IC50 = 60 nM T27137 C6MJB8 57908398 IC50 = 238 nM T27137 C1K3TI 57908399 IC50 = 190 nM T27137 C9UK4O 57908400 IC50 = 687 nM T27137 C4YVT6 57908404 IC50 = 4570 nM T27137 C8N4UB 60096231 EC50 > 25000 nM T27137 CG7K4H 60530531 EC50 < 10000 nM T27137 C4RD2I 67179855 IC50 = 65 nM T27137 CR84XZ 67180972 IC50 = 39 nM T27137 C4NG6L 67181122 IC50 = 92 nM T27137 C71SCP 67181213 IC50 = 100 nM T27137 CJ5G2L 67181693 IC50 = 67 nM T27137 CFM52I 67182239 IC50 = 7 nM T27137 CG0LC2 67182345 IC50 = 7 nM T27137 CBX67G 67246999 EC50 > 10000 nM T27137 CW7BI6 67424364 IC50 = 397 nM T27137 CA9LV5 67424813 IC50 = 1590 nM T27137 CC1HY4 67425269 IC50 = 735 nM T27137 C6M1FY 67425323 IC50 = 9540 nM T27137 C4LO1P 67425408 IC50 = 1020 nM T27137 C5JQ0F 67425734 IC50 = 2210 nM T27137 C5K7QG 67974411 EC50 > 10000 nM T27137 CCT07V 68290289 EC50 > 10000 nM T27137 C03JUE 68290572 EC50 > 10000 nM T27137 CQP9T0 70691553 IC50 = 110 nM T27137 CE85MJ 71455906 IC50 = 19 nM T27137 CO8D7T 71559536 IC50 = 891 nM T27137 C95DZX 71561287 IC50 = 1300 nM T27137 C2R4KC 71680758 IC50 = 398.11 nM T27137 CZD71P 71680760 IC50 = 97.72 nM T27137 CB35JV 71682339 IC50 = 2398.83 nM T27137 C1P3XF 71682340 IC50 = 161 nM T27137 CPHV98 71682341 IC50 = 977.24 nM T27137 CV1D9S 71682342 IC50 = 165.96 nM T27137 C8BO9P 71682343 IC50 > 30000 nM T27137 C8SG1R 71682344 IC50 > 30000 nM T27137 C0CVB7 71682491 IC50 > 30000 nM T27137 COA8H9 71682492 IC50 > 30000 nM T27137 C0L4EH 71682493 IC50 > 10000 nM T27137 C59JRI 71682494 IC50 > 31622.78 nM T27137 C0TBQ1 71682495 IC50 > 10000 nM T27137 CF1D4V 71682496 IC50 > 10000 nM T27137 CTQ16L 71682497 IC50 = 6606.93 nM T27137 CS4H1G 71682498 IC50 > 10000 nM T27137 CA4XT3 71682643 IC50 > 10000 nM T27137 C03QER 71682644 IC50 > 30000 nM T27137 CL0WC1 71682645 IC50 = 3610 nM T27137 C5WVU1 71682646 IC50 > 10000 nM T27137 CA4ZQ5 71682649 IC50 > 10000 nM T27137 CR2J9L 71682801 IC50 > 31622.78 nM T27137 CX69RU 71682802 IC50 = 596 nM T27137 CBC2D6 71682803 IC50 > 10000 nM T27137 CT68VQ 71682804 IC50 > 10000 nM T27137 C9WV8L 71682805 IC50 > 30000 nM T27137 CMK67X 71682806 IC50 = 707.95 nM T27137 C25DQG 71682958 IC50 > 10000 nM T27137 C0G7OV 71682959 IC50 = 1174.9 nM T27137 C1NMH0 71682960 IC50 > 10000 nM T27137 C64LHJ 71682961 IC50 = 1318.26 nM T27137 CSGC93 71682962 IC50 > 10000 nM T27137 CU0KW7 71682963 IC50 = 263.03 nM T27137 C0RLN1 71683123 IC50 = 2460 nM T27137 CCRO52 71683124 IC50 = 255 nM T27137 CLV85Q 71683125 IC50 = 416.87 nM T27137 CHJR06 71683126 IC50 = 707.95 nM T27137 CK9S3X 71683127 IC50 = 344 nM T27137 CVUJ25 71683128 IC50 = 1400 nM T27137 CAS1F0 71717012 IC50 > 12500 nM T27137 CXS25P 71717644 IC50 = 3110 nM T27137 CM10TY 71720053 IC50 > 12500 nM T27137 CSWB56 72163293 IC50 > 30000 nM T27137 C7CSF2 72163294 IC50 > 10000 nM T27137 CFA1K4 72163295 IC50 > 10000 nM T27137 C7XE3H 72163296 IC50 > 10000 nM T27137 C2IX5J 72163297 IC50 > 10000 nM T27137 CHP20F 72163298 IC50 = 5128.61 nM T27137 CG14IS 72163299 IC50 > 10000 nM T27137 CMI45T 72163300 IC50 > 30000 nM T27137 C6EC3O 72163432 IC50 = 85 nM T27137 C0M5CK 72163433 IC50 > 10000 nM T27137 CTY89D 72163434 IC50 = 1430 nM T27137 C6UM7X 72163435 IC50 > 10000 nM T27137 CD5WQ0 72163580 IC50 > 10000 nM T27137 CY2F8K 72163581 IC50 > 10000 nM T27137 C4VES7 72163582 IC50 = 676.08 nM T27137 CDJ03G 72163583 IC50 = 93 nM T27137 CB17ZM 72163584 IC50 = 478 nM T27137 C25SZK 72163585 IC50 = 1000 nM T27137 COZJ49 72163718 IC50 > 10000 nM T27137 CQ4HO9 72163719 IC50 = 185 nM T27137 CH6X1A 72163720 IC50 = 5590 nM T27137 CU17DE 72163721 IC50 = 831.76 nM T27137 C5Q3WO 72163722 IC50 > 10000 nM T27137 C9TX3E 72163723 IC50 = 549.54 nM T27137 CS5RI2 72163835 IC50 = 11748.98 nM T27137 CQ7CN8 72163836 IC50 > 10000 nM T27137 CNF81W 72163837 IC50 = 295.12 nM T27137 CVY58Q 72163838 IC50 = 769 nM T27137 CYT0Z7 72163839 IC50 = 363.08 nM T27137 CZ0G2X 72165213 IC50 = 30500 nM T27137 CXW8R2 72714783 EC50 > 10000 nM T27137 C6LT3X 73350553 IC50 > 10000 nM T27137 C91CBV 73350718 IC50 = 5128.61 nM T27137 C7N4GB 73350719 IC50 = 1905.46 nM T27137 CI51YQ 73355027 IC50 = 165.96 nM T27137 CIH73N 75238115 IC50 = 140 nM T27137 C4URX9 76310874 IC50 = 14000 nM T27137 C7LPF6 76318078 IC50 > 50000 nM T27137 COF43E 76321785 IC50 > 50000 nM T27137 CGV1R4 76321786 IC50 = 29800 nM T27137 C5BY7D 76325411 IC50 = 35700 nM T27137 CWJA51 76328955 IC50 = 5870 nM T27137 CTE1J7 76332628 IC50 > 50000 nM T27137 C80MQG 76332629 IC50 > 50000 nM T27137 CO0DA2 78320170 IC50 = 50 nM T27137 CQR1S8 78320479 IC50 = 499 nM T27137 CGU8O7 78320481 IC50 = 112 nM T27137 C61SXN 78320802 IC50 = 74 nM T27137 CEWF90 78320803 IC50 = 128 nM T27137 C5FP1U 78321115 IC50 = 57 nM T27137 C9OT3G 78321442 IC50 = 221 nM T27137 C43NLO 78322060 IC50 = 45 nM T27137 CZ0C4D 78322062 IC50 = 221 nM T27137 CKT06Q 78322063 IC50 = 747 nM T27137 C0UW2A 78322065 IC50 = 257 nM T27137 CRK06Y 78324865 IC50 = 136 nM T27137 C1LO8T 78324866 IC50 = 677 nM T27137 CZN2V7 78324867 IC50 = 58 nM T27137 CJF1S6 78324868 IC50 = 66 nM T27137 C4DR9A 78324869 IC50 = 407 nM T27137 CAZD45 78324870 IC50 = 374 nM T27137 C0ZT5H 78324871 IC50 = 162 nM T27137 C12ODV 86729801 IC50 = 184 nM T27137 CH4L7O 91885483 EC50 = 390 nM T27137 CJ5G3Q 118718091 EC50 = 3000 nM T27137 C8YQ7N 118735953 IC50 = 12200 nM T27137 C9XGN1 118735957 IC50 = 43200 nM T27137 C5SUP9 118735958 IC50 = 1420 nM T27137 C5NZX7 118735959 IC50 = 1090 nM T27137 C43QXF 118735961 IC50 = 2450 nM T27137 CCQ93P 118735962 IC50 = 2030 nM T27137 C71VQY 118735965 IC50 = 2820 nM T27137 C9E3CS 118735966 IC50 = 600 nM T27137 CV46AS 118735967 IC50 = 1240 nM T27137 CINE01 118735968 IC50 = 2900 nM T27137 C46HAM 118735969 IC50 = 4720 nM T27137 CXU1N4 118735970 IC50 = 3140 nM T27137 CZ6UX7 118735971 IC50 = 1810 nM T27137 CP3A6C 118735975 IC50 = 5310 nM T27137 CY8D9S 118735976 IC50 = 2380 nM T27137 CKZ02G 118735981 IC50 = 3090 nM T27137 CUC13P 122187795 IC50 > 30000 nM T27137 CU65XW 122193149 EC50 > 10000 nM T27137 CEC27S 122193150 EC50 > 10000 nM T27137 CEOP41 122193151 EC50 > 10000 nM T27137 CHEB16 122193152 EC50 > 10000 nM T27137 C7YVS5 122193153 EC50 < 10000 nM T27137 CM6WU5 122193154 EC50 = 4466.84 nM T27137 C1V0UA 122193155 EC50 < 10000 nM T27137 CG9QV2 122193156 EC50 > 10000 nM T27137 CK4M8L 122193157 EC50 < 10000 nM T27137 CF01PX 122193158 EC50 < 10000 nM T27137 C9VN6D 122193159 EC50 < 10000 nM T27137 C60PSU 122193160 EC50 < 10000 nM T27137 C6NBD3 122193161 EC50 > 10000 nM T27137 C6U3PF 122193162 EC50 > 10000 nM T27137 C74DFX 122193163 EC50 < 10000 nM T27137 CKV05E 122193164 EC50 < 10000 nM T27137 C1O5KH 122193165 EC50 > 10000 nM T27137 C1IFB2 122193166 EC50 > 10000 nM T27137 CH65KO 122193167 EC50 > 10000 nM T27137 C9AOE1 122193168 EC50 > 10000 nM T27137 C7Y1RV 122193169 EC50 > 10000 nM T27137 CW48QR 122193170 EC50 > 10000 nM T27137 C9I3LE 122193171 EC50 > 10000 nM T27137 C6JZ3S 122193172 EC50 < 10000 nM T27137 CMHP48 122193173 EC50 = 24.3 nM T27137 CE1L3P 122193174 EC50 = 54.4 nM T27137 CJIB74 122193175 EC50 = 33 nM T27137 C1N0HP 122193176 EC50 = 80.9 nM T27137 CV8J6N 122193177 EC50 = 31.8 nM T27137 C01PDA 122193178 EC50 = 23.99 nM T27137 CB8MH7 122193179 EC50 = 97.72 nM T27137 CK4IE1 122193310 EC50 = 291 nM T27137 CCP5U2 122195692 EC50 > 10000 nM T27137 CWHE41 122196091 IC50 = 47.86 nM T27137 CEG8I0 122196092 EC50 = 16 nM T27137 C2KA8E 122196093 EC50 = 29 nM T27137 C6TI1L 122196094 IC50 = 43.65 nM T27137 COC02R 122196095 EC50 = 22 nM T27137 CO48MD 122196096 EC50 = 26 nM T27137 CR34BM 122196097 EC50 = 28 nM T27137 CMUE28 122196098 EC50 = 35 nM T27137 C9WU0F 122196099 EC50 = 89 nM T27137 C2FI9X 122196100 EC50 = 21 nM T27137 C0BK2L 122196101 EC50 = 49 nM T27137 CS42ED 122196102 IC50 = 48.98 nM T27137 CPE1I5 122196103 EC50 = 123 nM T27137 CVIB23 122196104 EC50 = 530 nM T27137 CK2Z0Y 122196105 EC50 = 106 nM T27137 C5ODB4 122196106 IC50 = 154.88 nM T27137 CER92P 122196107 EC50 = 46 nM T27137 C4W6FN 122196108 EC50 = 49 nM T27137 C91DKH 122196109 EC50 = 18 nM T27137 CVFI45 122196110 EC50 = 144 nM T27137 CK6Q3M 122196111 EC50 = 387 nM T27137 CB7FN6 122196112 EC50 = 95 nM T27137 CZ08OD 122196113 EC50 = 35 nM T27137 C4VWT9 122196114 EC50 = 198 nM T27137 C65ABR 122196115 EC50 = 4610 nM T27137 CY9PM2 122196116 EC50 = 751 nM T27137 CRB9G8 122196117 EC50 = 208 nM T27137 CU7JC9 122196118 EC50 = 5330 nM T27137 CHT0B7 122196119 EC50 = 20 nM T27137 CZ0HS9 122196120 EC50 = 16 nM T27137 C7LP8W 122196121 IC50 = 22.39 nM T27137 CG5O4N 122196122 EC50 = 20 nM T27137 C2EXU4 122196123 IC50 = 12.59 nM T27137 CZ94FU 122196124 IC50 = 28.84 nM T27137 CM6T9O 122196125 EC50 = 15 nM T27137 CF8CV6 122196126 IC50 < 10000 nM T27137 C7PA4V 122196127 EC50 = 330 nM T27137 C2MK3Z 122196128 EC50 > 10000 nM T27137 CEV41Y 122196129 EC50 > 10000 nM T27137 CH2AO4 122539788 IC50 > 30000 nM T27137 CKIH28 127025478 EC50 > 10000 nM T27137 C2K9ZI 127025479 EC50 = 21.88 nM T27137 CYJD09 127025546 EC50 < 10000 nM T27137 CLO3T6 127025547 EC50 < 10000 nM T27137 C2XF0N 127025548 EC50 = 41 nM T27137 CIX4C9 127025549 EC50 = 469 nM T27137 CM56OW 127025550 EC50 = 1290 nM T27137 CX57FG 127025563 EC50 = 186.21 nM T27137 C7TVF2 127025564 EC50 = 251.19 nM T27137 CGYD41 127025831 EC50 = 141 nM T27137 CY9ZE6 127025845 EC50 < 10000 nM T27137 CH78CV 127025846 EC50 < 10000 nM T27137 CSXW80 127025847 EC50 = 673 nM T27137 C7FQ0Z 127025860 EC50 = 22.39 nM T27137 CECS36 127025861 EC50 > 10000 nM T27137 C47QGK 127026059 EC50 = 241 nM T27137 CDJ6A7 127026067 EC50 = 229.09 nM T27137 C0S2UW 127026137 EC50 = 1698.24 nM T27137 C1G5PU 127026138 EC50 = 50.12 nM T27137 CV3I2A 127026139 EC50 = 1370 nM T27137 CPB15M 127026140 EC50 = 63 nM T27137 CB2ZK5 127026165 EC50 = 11.48 nM T27137 C7J5VX 127026166 EC50 = 25.7 nM T27137 C9XU8I 127026167 EC50 = 5.37 nM T27137 CQ09MN 127026386 EC50 = 190.55 nM T27137 CFNI82 127026469 EC50 > 10000 nM T27137 CG8L6K 127026470 EC50 < 10000 nM T27137 CHJ2V0 127026471 EC50 = 557 nM T27137 CJH69G 127026472 EC50 = 851.14 nM T27137 C03DLS 127026473 EC50 > 10000 nM T27137 C82JTZ 127026474 EC50 = 630.96 nM T27137 C35SXQ 127027099 EC50 = 5248.07 nM T27137 C7QI9P 127027100 EC50 = 1890 nM T27137 CA42BO 127027101 EC50 = 19.5 nM T27137 C09CHL 127027102 EC50 = 22.39 nM T27137 CF2SH7 127027327 EC50 = 3420 nM T27137 CEDC20 127028298 EC50 = 263.03 nM T27137 CGJ86U 127028301 EC50 = 4365.16 nM T27137 C3SDP4 127028303 EC50 = 54 nM T27137 CRK8M7 127029000 EC50 = 1510 nM T27137 C24QVY 127029001 EC50 > 10000 nM T27137 C4QNP0 127029002 EC50 = 1470 nM T27137 CRV08S 127029301 EC50 = 56 nM T27137 CX4KF8 127029302 EC50 = 354.81 nM T27137 CH9XQ0 127029303 EC50 = 1230.27 nM T27137 COMY79 127030048 EC50 = 9549.93 nM T27137 CU8PT0 127030058 EC50 < 10000 nM T27137 CNJ65S 127030066 EC50 = 1130 nM T27137 CY23KD 127030339 EC50 < 10000 nM T27137 C89OKB 127030654 EC50 < 10000 nM T27137 CS2UY4 127030669 EC50 < 10000 nM T27137 C7A3ON 127030947 EC50 = 930 nM T27137 C3Y4UT 127030956 EC50 < 10000 nM T27137 CTYZ81 127030967 EC50 > 10000 nM T27137 CMQ36L 127031257 EC50 = 3715.35 nM T27137 CLF3J8 127031845 EC50 = 878 nM T27137 C7M6BT 127032498 EC50 < 10000 nM T27137 CIR78G 127032499 EC50 = 1760 nM T27137 CH9RF5 127032500 EC50 > 10000 nM T27137 C9UK1L 127032505 EC50 < 10000 nM T27137 C74TQG 127032506 EC50 = 484 nM T27137 C9G0AW 127032507 EC50 = 1070 nM T27137 C2A5HO 127032809 EC50 = 389.05 nM T27137 C3LC1K 127032838 EC50 > 10000 nM T27137 CX50VR 127032839 EC50 = 6520 nM T27137 CV14KJ 127033421 EC50 > 10000 nM T27137 CXV1P5 127033422 EC50 = 1258.93 nM T27137 C2B4JT 127033423 EC50 > 10000 nM T27137 CLTB96 127033424 EC50 = 1360 nM T27137 CGZ59R 127033432 EC50 = 1270 nM T27137 C4XJ8L 127033433 EC50 < 10000 nM T27137 CIA9E0 127033434 EC50 = 954 nM T27137 C3D7AY 127033435 EC50 = 4690 nM T27137 C7QL4E 127033436 EC50 = 223.87 nM T27137 CZ0P1G 127033437 EC50 = 3500 nM T27137 CK41TZ 127033693 EC50 = 5710 nM T27137 C3REZ4 127033694 EC50 = 3620 nM T27137 CE2NS9 127033724 EC50 > 10000 nM T27137 CIA5N4 127033725 EC50 < 10000 nM T27137 C3SU2D 127033960 EC50 = 2610 nM T27137 C01FRY 127033961 EC50 = 776.25 nM T27137 C9UER4 127033962 EC50 = 1318.26 nM T27137 C2POU1 127033963 EC50 = 177.83 nM T27137 CG0N2F 127034504 EC50 = 2090 nM T27137 CET40R 127034505 EC50 > 10000 nM T27137 C2QG3D 127034506 EC50 > 10000 nM T27137 C9A5VD 127034507 EC50 < 10000 nM T27137 CEQ1X9 127034512 EC50 = 6930 nM T27137 C03OAN 127034513 EC50 = 1548.82 nM T27137 C0L9UV 127034514 EC50 = 245 nM T27137 CKU1M0 127034515 EC50 = 353 nM T27137 C0A3DP 127034537 EC50 = 1290 nM T27137 C3X1IT 127046020 EC50 = 2691.53 nM T27137 CQCO27 127046038 EC50 = 219.28 nM T27137 C3S9JA 127047984 EC50 > 10000 nM T27137 C48NCK 127047993 EC50 = 180.6 nM T27137 C38BRY 131801162 EC50 > 10000 nM T27137 CFC05Q 131954513 IC50 > 10000000 nM T27137 C5YRP0 135659063 Ki = 6.7 nM T27137 CL2NW4 136244237 IC50 = 138 nM T27137 C3EGM5 137321168 IC50 > 10000 nM T27137 C3IL9H 155511336 IC50 > 30000 nM T27137 CYXE53 155538270 IC50 > 10000 nM T27137 CZ7NH0 155545491 IC50 > 30000 nM T27137 C29OSL 18003010 Ki = 4.8 nM T27137 D00EPM 73755217 IC50 > 30000 nM T27137 D00NCL 46836562 EC50 > 10000 nM T27137 D01ERW 11175501 IC50 = 3.5 nM T27137 D01EVA 6278000 IC50 = 3400 nM T27137 D01YEN 1233 Ki = 43000 nM T27137 D02NMN 23634102 IC50 = 2.1 nM T27137 D02NNU 16659803 IC50 = 2.2 nM T27137 D03NFW 11772954 IC50 = 3 nM T27137 D03OLR 71559428 IC50 = 409 nM T27137 D04DKM 104766 EC50 = 9300 nM T27137 D04JKL 2071 IC50 = 7000 nM T27137 D04MVR 11530404 IC50 = 3 nM T27137 D04RYE 46866192 IC50 = 27 nM T27137 D05DCW 46866191 IC50 = 2.1 nM T27137 D05KSC 11515548 IC50 = 43 nM T27137 D05NTV 10058919 IC50 = 68900 nM T27137 D05TFE 5218788 IC50 > 100000 nM T27137 D06DUE 40539 EC50 = 200 nM T27137 D06PAK 10058694 Ki > 100000 nM T27137 D06TYA 16659967 IC50 = 2.5 nM T27137 D07FXC 11299421 IC50 > 10000 nM T27137 D07GRG 10197984 Ki > 100000 nM T27137 D08CAB 83887 EC50 > 1000000 nM T27137 D08SCF 159548 IC50 = 23 nM T27137 D09AQK 4545574 Ki > 500000 nM T27137 D09QUN 58368068 EC50 > 10000 nM T27137 D09RPR 16737207 Ki > 10000 nM T27137 D09UBS 10428048 Ki > 100000 nM T27137 D0B3HH 9948645 Ki = 0.87 nM T27137 D0B4GX 9840951 IC50 = 28 nM T27137 D0D2GL 3972752 Ki > 1000000 nM T27137 D0DX6U 23725699 IC50 > 10000 nM T27137 D0EI9B 9903757 IC50 = 160 nM T27137 D0EK6P 5310984 Ki > 100000 nM T27137 D0G4BW 16659801 IC50 = 2.9 nM T27137 D0GX5C 16725048 IC50 = 7 nM T27137 D0H6BG 5866327 IC50 = 3000 nM T27137 D0IO8J 3025961 Ki = 36 nM T27137 D0J2WN 5311344 Ki > 270000 nM T27137 D0J8OW 446355 IC50 = 4300 nM T27137 D0L0YF 4236420 EC50 > 1000000 nM T27137 D0M2CT 9926999 IC50 = 96 nM T27137 D0N0NJ 15508178 IC50 > 300000 nM T27137 D0N2TF 10470232 IC50 = 14 nM T27137 D0N2TP 44190040 IC50 > 10000 nM T27137 D0N9UZ 9819927 Ki = 6800 nM T27137 D0O1AK 23327 EC50 > 1000000 nM T27137 D0O8WT 10338547 EC50 = 141.25 nM T27137 D0OH2P 5311040 IC50 = 25000 nM T27137 D0OS8Y 15985251 IC50 > 10000 nM T27137 D0OT9B 5960 EC50 > 1000000 nM T27137 D0OV2V 6324634 Ki > 300000 nM T27137 D0P3XO 5311459 IC50 = 58000 nM T27137 D0P6HX 11301185 IC50 = 3.6 nM T27137 D0PN6Z 179394 Ki > 1000000 nM T27137 D0Q6VH 5311432 IC50 > 100000 nM T27137 D0QC9F 16118537 IC50 = 12 nM T27137 D0R1YT 53316847 Ki = 0.4 nM T27137 D0R8EU 11245287 IC50 = 5.6 nM T27137 D0S6DK 5311455 IC50 = 40000 nM T27137 D0SB7U 57559562 IC50 = 6 nM T27137 D0SF9Z 16118119 IC50 = 6.3 nM T27137 D0SG6Q 23634171 IC50 = 0.9 nM T27137 D0T5SU 158397 EC50 > 1000000 nM T27137 D0U5YT 6604712 EC50 = 68000 nM T27137 D0V3YX 11537456 IC50 = 1 nM T27137 D0W0NJ 44442431 IC50 = 1412 nM T27137 D0W2GG 16659802 IC50 = 1.4 nM T98089 D0Z9QR 24066 Ki = 360000 nM T98089 D0D1LS 515328 IC50 > 4000 nM T98089 C0E8SU 64683 Ki = 1100000 nM T98089 CK40SL 24883191 IC50 = 1.7 nM T98089 C5SL1Q 25026090 IC50 = 10 nM T98089 CX6CE0 25026285 EC50 = 14 nM T98089 C6YOB7 25026288 IC50 = 38 nM T98089 CDU4W3 25026296 IC50 = 3600 nM T98089 CE8K6F 25026491 IC50 = 33 nM T98089 C0I3HQ 25026493 IC50 = 22 nM T98089 CG8AR2 25026495 EC50 = 13 nM T98089 CA3KO4 25026689 EC50 = 57 nM T98089 CB9WD4 25026690 EC50 = 36 nM T98089 CT6C1D 25026692 IC50 = 9 nM T98089 C91PIC 45375948 EC50 = 2 nM T98089 CF2H5G 45375949 IC50 = 2 nM T98089 C6D1KH 46846243 IC50 = 510 nM T98089 C14GNO 46879418 EC50 = 16000 nM T98089 CN1G5S 46879419 IC50 = 2700 nM T98089 C0NDG6 46879479 EC50 = 5500 nM T98089 CABJ15 46879480 EC50 = 2800 nM T98089 CP96AE 46879481 IC50 = 120 nM T98089 C1PWT4 46879482 IC50 = 110 nM T98089 CFY6R3 46879541 EC50 = 300 nM T98089 CO1PX5 46879542 IC50 = 49 nM T98089 CA0UQ3 46879543 IC50 = 63 nM T98089 CQ2ZG0 46879544 IC50 = 89 nM T98089 C0GSK6 46879584 EC50 = 13000 nM T98089 C9UL0C 46879585 IC50 = 15300 nM T98089 COUN32 46879586 IC50 = 51 nM T98089 C28MKP 46879587 IC50 = 79 nM T98089 CFV8X6 46879588 EC50 = 430 nM T98089 COA3I9 46879631 EC50 = 790 nM T98089 COV65T 46879632 EC50 = 160 nM T98089 CKGM61 46879633 IC50 = 95 nM T98089 CTVB71 46879634 EC50 = 530 nM T98089 C8NQS1 46879635 IC50 = 21 nM T98089 CZAH79 46879636 EC50 = 910 nM T98089 CX1DZ4 46879637 EC50 = 100 nM T98089 CT6O4N 46879671 IC50 = 5 nM T98089 CZ89PS 46879672 IC50 = 21 nM T98089 C86UTG 46879673 EC50 = 19 nM T98089 CGD0R8 46879674 EC50 = 270 nM T98089 C6R0QF 46879675 IC50 = 23 nM T98089 C03OXV 46879676 IC50 = 21 nM T98089 CUV71R 46879717 EC50 = 26 nM T98089 CFW93V 46879753 EC50 = 14 nM T98089 CO3AB1 46879754 EC50 = 61 nM T98089 C9PC3E 46879755 EC50 = 15 nM T98089 CQ2E7N 46879797 EC50 = 12 nM T98089 C45MBK 46879798 EC50 = 54 nM T98089 CUL9B5 46879799 EC50 = 140 nM T98089 C8Y9DS 46879855 IC50 = 5 nM T98089 C6ETK3 46879856 EC50 = 4 nM T98089 C9KVX6 46879857 EC50 = 13 nM T98089 C18SNL 46879892 EC50 = 20 nM T98089 C0DZ2R 46879893 EC50 = 5 nM T98089 C7PY3K 46879995 IC50 = 63 nM T98089 CS3BA2 60194750 Ki = 9.5 nM T98089 CQ90DI 60202339 IC50 = 37 nM T98089 CY0K9X 60202363 IC50 = 92 nM T98089 CR72NF 60202364 IC50 = 11 nM T98089 CCU9Z5 60202365 IC50 = 31 nM T98089 CIGP53 60202391 Ki = 0.5 nM T98089 CEA0M8 60202392 IC50 = 2.9 nM T98089 CU2X0Q 60202409 IC50 = 2.45 nM T98089 CFI0M9 60202411 IC50 = 1.07 nM T98089 CK4V0E 60202412 IC50 = 2.83 nM T98089 CB26HO 60202413 IC50 = 0.9 nM T98089 CI7F4Y 60202621 Ki = 1.5 nM T98089 CPFI60 60202622 IC50 = 150 nM T98089 C2F9NR 60202623 IC50 = 162 nM T98089 CK1S7Z 60202624 IC50 = 173 nM T98089 C5Z1GQ 60202625 IC50 = 230 nM T98089 CU0P7T 60202626 IC50 = 83 nM T98089 CL8D2X 71710912 Ki = 0.8 nM T98089 CPLX70 72706086 IC50 = 230 nM T98089 CRC17A 72706087 IC50 = 7 nM T98089 C9B4UR 73167565 Ki = 0.5 nM T98089 C5RK3I 73292701 Ki = 1.9 nM T98089 CB9VL8 73292702 IC50 = 8.01 nM T98089 CDM3E2 73292861 Ki = 8.9 nM T98089 CAE21Z 73292862 IC50 = 1.55 nM T98089 CNU2F0 73292863 IC50 = 2.85 nM T98089 C0C1RG 73292864 IC50 = 421 nM T98089 C0K9DS 73293026 IC50 = 534 nM T98089 C2SRZ1 73293027 IC50 = 506 nM T98089 CI46PU 73293028 IC50 = 251 nM T98089 CQ4V9R 73293029 IC50 = 512 nM T98089 CTXR32 73293030 IC50 = 1960 nM T98089 C8NUW3 73293031 IC50 = 1922 nM T98089 CJCK97 73293187 IC50 = 197 nM T98089 CBS64H 73293188 IC50 = 297 nM T98089 C93TOK 73293189 IC50 = 1041 nM T98089 C0QX6I 73293190 IC50 = 849 nM T98089 CGB90E 73293191 IC50 = 2367 nM T98089 CE8ST4 86223070 Ki = 735 nM T98089 C04SVT 86223073 Ki = 9.2 nM T98089 CKS2Z9 117889828 Ki = 6.8 nM T98089 CTM2O4 117890332 Ki = 1.8 nM T98089 CNQ76R 117890451 IC50 = 429.5 nM T98089 CLF5D7 117890462 IC50 = 10 nM T98089 CAB09G 118722637 Ki = 585 nM T98089 CXW7F6 118722638 IC50 = 1.25 nM T77645 CEL0O8 9833806 IC50 = 80 nM T77645 CNHD69 73347233 IC50 = 755 nM T77645 CF3B2T 73347234 IC50 = 3500 nM T69485 D00OVU 24965990 Ki = 0.35 nM T69485 D06CKX 25195495 Ki = 0.3981 nM T69485 D08SCL 46190695 Ki = 1.1 nM T69485 D0A7ZK 56944144 Ki = 0.44 nM T69485 D0FK6O 67116280 Ki = 9 nM T69485 D0NN5A 25128145 Ki = 0.1995 nM T69485 D06BTF 23727689 Ki = 4.7 nM T69485 C91DAE 185394 IC50 = 900 nM T69485 CKN27R 645882 Ki = 1000 nM T69485 CW90GD 647720 Ki = 100 nM T69485 CMQ23R 833756 Ki > 10000 nM T69485 C5NO3B 855282 Ki > 15848.93 nM T69485 C1Q7FH 1034375 IC50 = 130 nM T69485 CCN92H 1207917 IC50 = 500 nM T69485 CEX5I0 1301005 IC50 = 10 nM T69485 CK8ZP2 1725151 IC50 = 346 nM T69485 C7L9OX 1784975 IC50 > 10000 nM T69485 CZ0AJ2 2273636 IC50 = 232 nM T69485 CDC1E3 2796191 Ki = 25 nM T69485 CC79VB 2860019 IC50 = 70 nM T69485 C4JH3Z 2870209 IC50 = 1700 nM T69485 CV53JP 3119056 IC50 = 19 nM T69485 CF8RB9 3119749 IC50 = 800 nM T69485 CG01OM 3213606 Ki = 1000 nM T69485 C4X9CJ 3213619 Ki = 1584.89 nM T69485 C4XGO6 3213626 Ki = 39.81 nM T69485 C8WE7J 3213637 Ki > 15848.93 nM T69485 CL6KP4 3213649 Ki = 50.12 nM T69485 C89CAQ 3213663 Ki > 15848.93 nM T69485 C7XRC5 3213671 Ki = 2.512 nM T69485 CA9E7M 3213679 Ki > 15848.93 nM T69485 CL7PN8 3213689 Ki = 501.19 nM T69485 CFPR85 3213696 Ki = 1.585 nM T69485 CLX9G8 3213712 Ki = 199.53 nM T69485 C9L6CG 3213744 Ki = 15.85 nM T69485 CU8F4X 3213776 Ki = 31.62 nM T69485 CJ93NE 3213793 Ki = 501.19 nM T69485 CHS5V2 3213803 Ki = 1995.26 nM T69485 C4O1NG 3213835 Ki = 100 nM T69485 C0IW7Z 3213904 Ki = 398.11 nM T69485 C3XD5Z 3213915 Ki = 501.19 nM T69485 CM2S1K 3213928 Ki = 158.49 nM T69485 C32UAN 3213941 Ki > 15848.93 nM T69485 C5R4LA 3213958 Ki = 158.49 nM T69485 CYM81H 3213966 Ki = 63.1 nM T69485 C8XAM0 3213992 Ki = 39.81 nM T69485 CS0VF3 3214024 Ki = 316.23 nM T69485 C2J1TB 3634416 IC50 = 700 nM T69485 C3O5WZ 5165198 Ki = 398.11 nM T69485 C04ZBY 5218889 IC50 = 700 nM T69485 CT23BD 6418917 IC50 = 300 nM T69485 CX1BS0 6859582 IC50 = 11800 nM T69485 CTYZ64 9798764 Ki = 1704 nM T69485 C7SN9C 9936247 IC50 = 36 nM T69485 CR3LK5 9978819 Ki = 79.43 nM T69485 C2ELV0 9978820 Ki = 50.12 nM T69485 CK0F1B 10024157 Ki = 1584.89 nM T69485 C25NXP 10024223 Ki = 1000 nM T69485 CR4VC2 10044549 Ki = 2511.89 nM T69485 C8TZF9 10046197 Ki = 63.1 nM T69485 CO41BA 10046198 Ki < 5011.87 nM T69485 CER65W 10048862 Ki = 6.31 nM T69485 CC0V9S 10069829 Ki = 251.19 nM T69485 C8SHP4 10112247 IC50 > 10000 nM T69485 C7UL5G 10113123 Ki = 4 nM T69485 C8MS0F 10139334 IC50 = 1161 nM T69485 C41SAC 10144095 IC50 = 240 nM T69485 C5CZ0J 10201185 Ki = 19.95 nM T69485 CV0Y8N 10204153 Ki = 129 nM T69485 CVN2Q8 10208109 IC50 > 10000 nM T69485 C46ROY 10250023 Ki = 100 nM T69485 CTHA73 10278102 IC50 = 8152 nM T69485 C69ZAN 10316124 Ki = 125.89 nM T69485 CYB3G4 10316232 Ki = 2511.89 nM T69485 CQNX31 10316508 Ki = 79.43 nM T69485 CWU80C 10337554 Ki = 398.11 nM T69485 CJSX37 10386388 Ki = 100 nM T69485 CZS4R9 10387337 Ki = 39.81 nM T69485 C8OF7V 10407090 Ki = 63.1 nM T69485 CA3E0X 10409682 IC50 = 5 nM T69485 C4E9ZR 10433189 Ki = 79.43 nM T69485 C3LJ1G 10453273 Ki = 19.95 nM T69485 C5FBU7 10473775 Ki = 1584.89 nM T69485 CZ1J7A 10475401 IC50 = 89 nM T69485 CX7M8O 10864072 IC50 = 2686 nM T69485 C7OM4V 10864264 IC50 = 14 nM T69485 CBM0E3 10864538 IC50 = 101 nM T69485 CUPD25 10874416 IC50 > 10000 nM T69485 CV83MQ 10884498 IC50 = 6103 nM T69485 C8ZEK0 10906648 IC50 > 10000 nM T69485 CKV5W9 10918096 IC50 > 10000 nM T69485 C2VF5E 10918199 IC50 = 80 nM T69485 CVI01B 10929426 IC50 = 19 nM T69485 C0MWO4 10939830 IC50 = 4198 nM T69485 CVG1W4 10939855 IC50 = 5660 nM T69485 CKNF23 10951393 IC50 = 679 nM T69485 C4ZTW3 10951496 IC50 = 109 nM T69485 C8E5LJ 10962350 IC50 = 1098 nM T69485 CE68HD 10983971 IC50 = 9499 nM T69485 CADV49 10983972 IC50 = 10000 nM T69485 CRNI02 10994188 IC50 > 10000 nM T69485 CR9S3I 10994415 IC50 = 10000 nM T69485 C9KAL2 11016474 IC50 > 10000 nM T69485 C5W8OD 11016554 IC50 = 281 nM T69485 CC0IG1 11038242 IC50 > 10000 nM T69485 C4DX9L 11049263 IC50 = 10000 nM T69485 C3NL0R 11071336 IC50 = 1536 nM T69485 CZF1P3 11071351 IC50 = 10000 nM T69485 C47DCI 11081493 IC50 = 10000 nM T69485 C8RK9Q 11081686 IC50 = 10000 nM T69485 CF9D3V 11102681 IC50 > 10000 nM T69485 C5G1WK 11123332 IC50 > 10000 nM T69485 CGA21K 11146397 IC50 = 1814 nM T69485 CM26ZQ 11734173 IC50 = 1811 nM T69485 C6KE0W 11744563 Ki = 79.43 nM T69485 CZ0TU8 11812976 IC50 = 10000 nM T69485 CM6A3U 11960895 Ki = 0.2 nM T69485 CHV29L 11960929 Ki = 4 nM T69485 CQD14I 12047522 IC50 > 10000 nM T69485 C5SR3I 12997499 IC50 = 910 nM T69485 CXGJ06 15949515 Ki = 3 nM T69485 CDXM06 15949516 Ki = 2 nM T69485 CBF2K7 15949607 Ki = 6 nM T69485 C1EIU3 15949609 Ki = 11 nM T69485 CA3C9D 15949610 Ki = 1 nM T69485 C9V6OR 15949701 Ki = 280 nM T69485 C75IUA 15949702 Ki = 11 nM T69485 CM61GE 15949703 Ki = 3 nM T69485 CJ4X8D 15993497 IC50 = 661 nM T69485 C52SLH 16002587 Ki > 10000 nM T69485 C81AUJ 16046844 Ki = 15.85 nM T69485 C0BLR7 16048438 Ki = 186.21 nM T69485 C9RM2Y 16752731 IC50 = 4 nM T69485 CKH6B4 18592212 Ki = 0.7943 nM T69485 CK7L1A 18592214 Ki = 25.12 nM T69485 CT6ON8 18592216 Ki = 79.43 nM T69485 CJBK87 20911062 IC50 = 35 nM T69485 CQE54R 22599910 IC50 = 2100 nM T69485 CW7F3D 22599915 IC50 = 900 nM T69485 CKL08P 22599923 IC50 > 10000 nM T69485 CIO42U 24737677 IC50 = 5 nM T69485 CBC56J 24748750 IC50 = 6 nM T69485 CH6TN9 24759955 IC50 = 5 nM T69485 CY3X7G 24760024 IC50 = 7 nM T69485 C4R8OV 24760087 IC50 = 4.5 nM T69485 C9B2DL 24760747 IC50 = 5 nM T69485 C43PRK 24760748 IC50 = 10 nM T69485 CB3TQ1 24808511 IC50 = 50 nM T69485 C1H3AN 24808514 Ki = 0.17 nM T69485 CK5LN1 24853522 IC50 = 24 nM T69485 COB2P9 24882716 Ki = 0.59 nM T69485 CB9SA1 24896566 Ki = 0.7 nM T69485 CZ9EQ2 24959177 IC50 = 9 nM T69485 C9MI0U 24959178 IC50 = 8 nM T69485 CJR42H 24959549 IC50 = 7 nM T69485 CY58BS 24959912 IC50 = 12 nM T69485 C50TAB 24960290 IC50 = 11 nM T69485 C5UF2L 24960654 IC50 = 11 nM T69485 CTE96G 24961018 IC50 = 23 nM T69485 CUI6E1 24961746 IC50 = 18 nM T69485 C35DNF 24961747 IC50 = 17 nM T69485 C67KNQ 24962111 IC50 = 18 nM T69485 C57LWU 24962112 IC50 = 16 nM T69485 CG43WT 24962115 IC50 = 60 nM T69485 CK9H5Y 24962833 IC50 = 9 nM T69485 CL6N8O 24962835 IC50 = 4 nM T69485 CCGY36 24964221 Ki = 6.3 nM T69485 C95RZN 24964358 Ki = 3500 nM T69485 C8XHN9 24964574 Ki = 11 nM T69485 C9IUP7 24964576 Ki = 3.7 nM T69485 C38UID 24964578 Ki = 0.5 nM T69485 CYEP21 24964937 Ki = 0.2 nM T69485 CTX7I1 24964940 Ki = 1.5 nM T69485 CV58CQ 24965286 Ki = 1.6 nM T69485 CW7S0O 24965287 Ki = 0.7 nM T69485 C5I9DX 24965290 Ki = 0.6 nM T69485 C5SFH2 24965291 Ki = 1.2 nM T69485 CGP45R 24965643 Ki = 0.28 nM T69485 CSI6H9 24965645 Ki = 0.25 nM T69485 CFS95W 24968277 Ki = 0.9 nM T69485 CPQD14 24992490 IC50 = 13 nM T69485 CTI38U 25060119 Ki = 0.07 nM T69485 CTX03U 25060120 Ki = 78.5 nM T69485 C8XKP2 25060382 Ki = 40.5 nM T69485 CXE52R 25060383 Ki = 18 nM T69485 CD6CA4 25060384 Ki = 22 nM T69485 C6L1VC 25060653 Ki = 4.1 nM T69485 C8DO2L 25060654 Ki = 3 nM T69485 CN7V6R 25060655 Ki = 4.8 nM T69485 C0K6WX 25060657 Ki = 0.6 nM T69485 C5U9ZY 25060899 Ki = 0.8 nM T69485 CDBQ73 25060900 Ki = 8.3 nM T69485 C56RMG 25060902 Ki = 1.3 nM T69485 CMOS06 25063585 IC50 = 6 nM T69485 CF5AB2 25063587 IC50 = 7 nM T69485 CJY0H7 25063628 IC50 = 12 nM T69485 C7ZP8R 25063664 IC50 = 19 nM T69485 C9KY3W 25063665 IC50 = 21 nM T69485 C39RAF 25063701 IC50 = 22 nM T69485 C92NVF 25110749 IC50 = 25.12 nM T69485 C1CFZ4 25110750 IC50 < 30 nM T69485 CS31WP 25110751 IC50 < 30 nM T69485 CO47QV 25127474 IC50 = 562.34 nM T69485 C15XCU 25127493 Ki = 0.2 nM T69485 CY5X1A 25204740 IC50 = 18 nM T69485 C03XSU 25225718 Ki = 0.3 nM T69485 CF5MV8 25809483 IC50 = 195 nM T69485 C07DOP 26719840 IC50 = 7 nM T69485 CW2U6O 30560665 IC50 = 96 nM T69485 CYL39Q 40924317 Ki = 0.631 nM T69485 C7IKX4 42604859 Ki = 1.1 nM T69485 CT13OI 44219762 Ki = 2 nM T69485 CI4BE6 44270595 EC50 > 1000000 nM T69485 CW30VO 44270596 EC50 > 1000000 nM T69485 C26BKD 44270597 EC50 > 1000000 nM T69485 C39TRO 44270625 EC50 > 1000000 nM T69485 C5PO4S 44270635 EC50 > 1000000 nM T69485 C87IBU 44270666 EC50 > 1000000 nM T69485 CMB6A1 44270673 EC50 > 1000000 nM T69485 C1OM8C 44270674 EC50 > 1000000 nM T69485 CZW96I 44270676 EC50 > 1000000 nM T69485 CQ56DO 44270709 EC50 > 1000000 nM T69485 C6GJW8 44359225 IC50 = 28 nM T69485 CUPE16 44359281 IC50 = 35 nM T69485 C68CJQ 44359282 IC50 = 25 nM T69485 C9H4QW 44359283 IC50 = 59 nM T69485 C5FKZ8 44359335 IC50 > 10000 nM T69485 CQP59C 44359365 IC50 = 70 nM T69485 CIO8P6 44359366 IC50 = 2900 nM T69485 CE4FG6 44359367 IC50 = 130 nM T69485 C7SO5Y 44359405 IC50 > 10000 nM T69485 CCG51L 44359415 IC50 = 56 nM T69485 CX4C8G 44359451 IC50 > 10000 nM T69485 CSY89K 44359452 IC50 = 3300 nM T69485 CA31JT 44359467 IC50 > 10000 nM T69485 C9YK1T 44359482 IC50 = 240 nM T69485 CFJI51 44359494 IC50 > 10000 nM T69485 COVU19 44359603 IC50 = 1400 nM T69485 CUQ13D 44359613 IC50 = 30 nM T69485 CN73FK 44359637 IC50 = 2000 nM T69485 CR9E8A 44359650 IC50 = 395 nM T69485 C9QD1O 44376981 EC50 = 947 nM T69485 CD62VI 44393273 Ki = 398.11 nM T69485 C47MUJ 44393285 Ki = 316.23 nM T69485 CT3U9Z 44393313 Ki = 25.12 nM T69485 C5QNK7 44393337 Ki = 199.53 nM T69485 CIWP10 44393338 Ki = 199.53 nM T69485 C81EBC 44393370 Ki = 501.19 nM T69485 C4X2QA 44393375 Ki = 1258.93 nM T69485 CH0UI9 44405008 EC50 = 0.72 nM T69485 CM1IS8 44454577 Ki = 0.6 nM T69485 CA39CP 44454599 Ki = 560 nM T69485 C1BD8E 44454602 Ki = 131 nM T69485 CR35JH 44454877 Ki = 0.8 nM T69485 C9OD7E 44454878 Ki = 0.1 nM T69485 CLRZ97 44454915 Ki = 0.09 nM T69485 CZG78N 44454916 Ki = 8 nM T69485 CYIO02 44454917 Ki = 0.2 nM T69485 CSLE81 44454943 Ki = 2 nM T69485 CWPB72 44454946 Ki = 0.3 nM T69485 C2RO9B 44454947 Ki = 2 nM T69485 C3I1LF 44463491 Ki = 63.1 nM T69485 CJY9N1 44555825 IC50 = 2 nM T69485 C92PMB 44555872 IC50 = 1 nM T69485 C2JT5F 44555974 IC50 = 14 nM T69485 C9UH1P 44555976 IC50 = 25 nM T69485 C7P2VN 44555978 IC50 = 9 nM T69485 CJU9R7 44556023 IC50 = 26 nM T69485 C38KGZ 44556024 IC50 = 7 nM T69485 C3A8UM 44563904 IC50 = 17 nM T69485 C3IA9R 44563928 IC50 = 4 nM T69485 CCRY94 44563929 IC50 = 2 nM T69485 C5ASO0 44564034 IC50 = 28 nM T69485 CR0T4G 44564035 IC50 = 10000 nM T69485 CQ6Y4K 44564036 IC50 = 10000 nM T69485 CFA0L2 44564038 IC50 = 36 nM T69485 C7R9DP 44574230 Ki = 550 nM T69485 CZQ2N6 44574255 Ki = 240 nM T69485 C7IYO9 44574256 Ki = 120 nM T69485 C67JEM 44574257 Ki = 42 nM T69485 CUZK61 44580808 IC50 = 139 nM T69485 C2R8YC 44580809 IC50 = 839 nM T69485 C0LDE2 44580810 IC50 = 463 nM T69485 CHIG04 44580825 IC50 = 48 nM T69485 C6HQ2K 44580862 IC50 = 239 nM T69485 CLP6W7 44580863 IC50 = 110 nM T69485 C0BJI8 44580864 IC50 = 789 nM T69485 CLKU70 44580865 IC50 = 4 nM T69485 C5INH4 44580886 IC50 = 60 nM T69485 C2HT8N 44580887 IC50 = 8 nM T69485 CUM2B9 44580888 IC50 = 90 nM T69485 C3FSE5 44580889 IC50 = 2405 nM T69485 CJ3HV2 44580912 IC50 = 433 nM T69485 CEB05Y 44580913 IC50 = 1606 nM T69485 CC8D7N 44580914 IC50 = 1161 nM T69485 CY0A2T 44580945 IC50 = 5 nM T69485 CR8EL1 44580946 IC50 = 3 nM T69485 C2O6MI 44580947 IC50 = 7 nM T69485 CA36HG 44580948 IC50 = 4 nM T69485 CE4UV6 44580968 IC50 = 5 nM T69485 CVMS64 44580969 IC50 = 7 nM T69485 CNUF76 44581140 IC50 = 142 nM T69485 CHZO78 44581141 IC50 = 1187 nM T69485 COUS06 44581168 IC50 = 1822 nM T69485 CNK67Y 44581169 IC50 = 58 nM T69485 CZ03FY 44581170 IC50 = 800 nM T69485 C41ZJE 44581171 IC50 = 3372 nM T69485 C97LXJ 44581172 IC50 = 60 nM T69485 C5OYV4 44589638 IC50 = 302 nM T69485 CQH96O 44589674 IC50 = 229.09 nM T69485 CD24QJ 44589675 IC50 = 323.59 nM T69485 CG1C2A 44589711 IC50 = 109.65 nM T69485 C0O6IX 44589712 IC50 = 151.36 nM T69485 CHWI96 44589748 IC50 = 138.04 nM T69485 C64IJQ 44589749 IC50 = 81.28 nM T69485 CBP2Z4 44589750 IC50 = 194.98 nM T69485 C5Z2VB 44589751 IC50 = 51.29 nM T69485 C2L4WI 44589787 IC50 = 107.15 nM T69485 CL3BG5 44589788 IC50 = 131.83 nM T69485 C1SYK4 44633765 Ki = 0.5 nM T69485 CRM6C5 45259003 Ki = 0.3 nM T69485 C1QS3Y 45259004 Ki = 2.1 nM T69485 CH97EI 45375925 Ki = 0.9 nM T69485 COF2A8 45501596 Ki = 251.19 nM T69485 CMRT28 45555989 IC50 = 710 nM T69485 CB4O9P 46190694 Ki = 0.5 nM T69485 C3KB9Q 46191662 Ki = 1.4 nM T69485 CRM02K 46191726 Ki = 7.6 nM T69485 CBGP17 46191727 Ki = 10 nM T69485 CJK6P2 46195690 Ki = 0.3 nM T69485 CSJ27E 46204871 Ki = 1.4 nM T69485 CI34NU 46205522 Ki = 8.3 nM T69485 C2U1KF 46211807 Ki = 9.8 nM T69485 C0LQ6S 46211878 Ki = 9.3 nM T69485 C51BQE 46211883 Ki = 7.5 nM T69485 C48TNW 46211956 Ki = 6.8 nM T69485 C21ICG 46212134 Ki = 0.6 nM T69485 C8R3SM 46212185 Ki = 1.3 nM T69485 CFV4Q2 46212296 Ki = 0.24 nM T69485 CHD1J4 46212539 Ki = 5.1 nM T69485 CO7N9S 46212746 Ki = 621 nM T69485 CT6F9H 46868664 Ki = 0.36 nM T69485 CNJR98 46868665 Ki = 0.47 nM T69485 CRK9B5 46868791 Ki = 3.2 nM T69485 C1KRZ6 46868793 Ki = 8.5 nM T69485 C7DH6F 46880346 IC50 = 219 nM T69485 CP4C1B 46880347 IC50 = 3 nM T69485 C9Y3QE 46880348 IC50 = 174 nM T69485 CMPE07 46880349 IC50 = 9 nM T69485 CJBC31 46880388 IC50 = 179 nM T69485 CZ3C8T 46880389 IC50 = 10 nM T69485 C8ECV5 46880449 IC50 = 3 nM T69485 C29IMV 46880450 IC50 = 19 nM T69485 C6JK5G 46880451 IC50 = 25 nM T69485 CFX08U 46883808 Ki = 0.2 nM T69485 C9C0FR 46883864 Ki = 11 nM T69485 CFL51W 46883865 Ki = 260 nM T69485 CR56NI 46883908 Ki = 0.6 nM T69485 CH5M1P 49793266 Ki = 1.4 nM T69485 C51JSQ 49797987 Ki = 0.4 nM T69485 CS19WL 49797988 Ki = 0.8 nM T69485 CS9WK7 49798002 Ki = 2.9 nM T69485 C39KIH 49798003 Ki = 62 nM T69485 CR0C5N 49798004 Ki = 105 nM T69485 CNV6E4 49798005 Ki = 590 nM T69485 C3F0HR 49798028 Ki = 2.2 nM T69485 C72ADP 49798029 Ki = 14 nM T69485 C1X8TR 49798030 Ki = 0.6 nM T69485 C2BS3P 49805788 IC50 = 16 nM T69485 C0DKB7 50799599 Ki = 78 nM T69485 CS1O7E 52918933 Ki = 12 nM T69485 C51EGW 52942033 Ki = 630.96 nM T69485 C65JKN 52944312 Ki = 1000 nM T69485 CFC12V 52944709 Ki = 398.11 nM T69485 C9X3BC 52946457 Ki = 251.19 nM T69485 CY9JU2 52948927 Ki = 1995.26 nM T69485 CJ4S2D 53242191 Ki = 61.66 nM T69485 CCZL67 53242213 Ki = 3 nM T69485 C8TC5B 53259112 Ki = 77.62 nM T69485 C68ERM 53259279 Ki = 181.97 nM T69485 CK5CM6 53259467 Ki = 25 nM T69485 C6U4FE 53259634 Ki = 12.88 nM T69485 CXKZ15 53259635 Ki = 3.162 nM T69485 C1HT7I 53259636 Ki = 69.18 nM T69485 C5E6TF 54576281 Ki = 5.7 nM T69485 CI64JB 54579367 IC50 = 1 nM T69485 CUG05N 54579583 IC50 = 0.8 nM T69485 CAG6V1 54579585 IC50 = 194 nM T69485 CLT6O5 54588789 IC50 = 14 nM T69485 C0OIE7 54751924 IC50 = 27 nM T69485 C96GZT 54765113 Ki = 417 nM T69485 CA0YR4 56659966 Ki = 19.95 nM T69485 CC6M4B 56663428 Ki = 1258.93 nM T69485 CK76VA 56663429 Ki = 31.62 nM T69485 CU84LF 56670285 Ki = 501.19 nM T69485 C37HIB 56673796 Ki > 3162.28 nM T69485 C3CO2F 56673797 Ki = 125.89 nM T69485 CPT8J3 56673798 Ki = 5.012 nM T69485 CPE3R9 56680444 Ki = 630.96 nM T69485 C5TY1F 56680445 Ki = 19.95 nM T69485 CG6D7M 56680446 Ki = 31.62 nM T69485 CC0QF6 56683774 Ki = 0.7943 nM T69485 C35PTG 56683775 Ki = 0.2512 nM T69485 CW80YF 56943752 Ki = 7 nM T69485 CP5UD4 56944043 Ki = 4 nM T69485 C6F3VI 56944044 Ki = 7 nM T69485 CU87RH 56944045 Ki = 2 nM T69485 C67OXC 56944143 Ki = 2 nM T69485 C0BKG3 56944244 Ki = 5 nM T69485 C6GDX1 56944245 Ki = 8 nM T69485 CNY8F7 56944337 Ki = 7 nM T69485 C09WRF 56944429 Ki = 3 nM T69485 CAP79V 56944521 Ki = 9 nM T69485 C3SY9G 56944522 Ki = 1 nM T69485 CJ5T0W 56944620 Ki = 1 nM T69485 CX41CZ 56968452 Ki = 6.918 nM T69485 C6RH9Z 56970209 Ki = 17.38 nM T69485 CZQ5T1 56970417 Ki = 7 nM T69485 C7I0LP 56970421 Ki = 0.7 nM T69485 C15GZB 56970625 Ki = 20.89 nM T69485 CB4F3T 56970626 Ki = 0.8511 nM T69485 CF7M3A 56970628 Ki = 6.918 nM T69485 CRV8S0 56970857 Ki = 26.92 nM T69485 CDIO92 56970858 Ki = 14.13 nM T69485 CK9SF5 57388373 Ki > 2000 nM T69485 C56ORS 57388650 Ki = 5 nM T69485 CYQ43V 57388812 IC50 = 51.7 nM T69485 C1DF3J 57389725 IC50 = 2.81 nM T69485 CF08CS 57389801 IC50 = 11.9 nM T69485 CKDI91 57389883 IC50 = 198 nM T69485 C4FC6Z 57390049 IC50 = 14.2 nM T69485 C2LTP8 57390051 IC50 = 1460 nM T69485 CO7MP1 57390997 IC50 = 160 nM T69485 CB4CA1 57391006 IC50 = 230 nM T69485 C23QDY 57391099 IC50 = 430 nM T69485 C29SFQ 57392779 IC50 = 6400 nM T69485 CAPD05 57392800 IC50 = 130 nM T69485 C4AR0T 57392874 IC50 = 4700 nM T69485 CLV50P 57392875 IC50 = 730 nM T69485 CY6XR2 57394509 IC50 = 150 nM T69485 C5WV2G 57396272 IC50 = 87 nM T69485 CI43RF 57396356 IC50 = 6.4 nM T69485 COF59D 57396357 IC50 = 140 nM T69485 C8DY2G 57398059 IC50 = 74 nM T69485 C3Y6HM 57398157 IC50 = 3000 nM T69485 C48ROC 57398158 IC50 = 270 nM T69485 C4BY0H 57401580 IC50 = 8200 nM T69485 C0K1PV 57403243 IC50 = 1000 nM T69485 C40IOT 57403244 IC50 = 3.3 nM T69485 C9NHI3 58394291 Ki = 4.5 nM T69485 CXA3T8 58488153 Ki = 39 nM T69485 CI7U5V 60168601 IC50 = 1.4 nM T69485 CE9IM4 66733985 IC50 = 227 nM T69485 C8XNW4 67153780 IC50 = 10 nM T69485 CXQ94P 67153782 IC50 = 35 nM T69485 C5FN3I 67209228 Ki = 527 nM T69485 C4PGT2 67209346 Ki = 2 nM T69485 CX2F3S 67209359 Ki = 158 nM T69485 CC2IT1 67209405 Ki = 26 nM T69485 CB7W0G 67209575 Ki = 582 nM T69485 C69PEQ 67209610 Ki = 83 nM T69485 C0C4JF 67209817 Ki = 59 nM T69485 CU5C8L 67251476 Ki = 588.84 nM T69485 CC6X2O 67252378 Ki = 0.4571 nM T69485 C4KC6Q 67281908 Ki = 6 nM T69485 CZ4L7E 67282493 Ki = 2 nM T69485 C3Q6ZA 67282848 Ki = 4 nM T69485 C4R1IH 67283149 Ki = 4 nM T69485 C0S7IR 67289227 Ki = 3.89 nM T69485 C15EQH 67380581 Ki = 28.9 nM T69485 CH6EW0 67473922 Ki = 29 nM T69485 C1I7OW 67473934 Ki = 80 nM T69485 CK18IT 67473935 Ki = 50 nM T69485 C2VD6Q 67473936 Ki = 163 nM T69485 C42FLR 67473937 Ki = 56 nM T69485 CK1Q3V 67473938 Ki = 34 nM T69485 C2D4VM 67980311 Ki = 5 nM T69485 C0U9GM 67980666 Ki = 36 nM T69485 CEVG41 68058790 Ki = 222 nM T69485 CDQ31I 68058793 Ki = 21 nM T69485 CTL92R 68083077 Ki = 17 nM T69485 CW8FR2 69080080 IC50 = 507 nM T69485 CUIC59 69080156 IC50 = 34 nM T69485 CCB80U 69080186 IC50 = 133 nM T69485 CV4NO2 69080188 IC50 = 128 nM T69485 CN5H2Z 69080268 IC50 = 252 nM T69485 C58BVC 69080890 IC50 = 74 nM T69485 CE4I3Q 69080992 IC50 = 37 nM T69485 CJ7VG2 69081444 IC50 = 6 nM T69485 C49PMK 69081570 IC50 = 8 nM T69485 CNJ7K2 69081619 IC50 = 168 nM T69485 C4IW9J 69081640 IC50 = 41 nM T69485 CU4Z7I 69081642 IC50 = 894 nM T69485 CY0K1B 69081717 IC50 = 25 nM T69485 CD8RY3 69081742 IC50 = 9 nM T69485 CI3M2O 69081821 IC50 = 21 nM T69485 CSX60D 69081873 IC50 = 28 nM T69485 C30PMS 69081899 IC50 = 1291 nM T69485 CJI32G 69081964 IC50 = 329 nM T69485 CIN3O2 69082001 IC50 = 3610 nM T69485 C3RDA0 69082236 IC50 = 19 nM T69485 C0QY5T 69082267 IC50 = 635 nM T69485 CUW42P 69082306 IC50 = 47 nM T69485 C72OGM 69082473 IC50 = 268 nM T69485 CJ93CT 69082475 IC50 = 12 nM T69485 C8L6DC 69082510 IC50 = 6 nM T69485 C6QB2K 69082516 IC50 = 2 nM T69485 CHS32F 69082545 IC50 = 6940 nM T69485 C95XAQ 69082595 IC50 = 670 nM T69485 CNK12W 69082599 IC50 = 589 nM T69485 CW6MR8 69082645 IC50 = 119 nM T69485 C61XNT 69082665 IC50 = 154 nM T69485 CD5HB2 69082678 IC50 = 563 nM T69485 CV94BF 69082681 IC50 = 1002 nM T69485 CLX8D3 69082742 IC50 = 42 nM T69485 CJ45VT 69082766 IC50 = 86 nM T69485 CB70SA 69082817 IC50 = 94 nM T69485 COE39Z 69082854 IC50 = 59 nM T69485 C96STB 69082926 IC50 = 93 nM T69485 C6PR7O 69083435 IC50 = 133 nM T69485 CQ1IK8 69083745 IC50 = 161 nM T69485 CPLG25 69083777 IC50 = 4 nM T69485 CJ6A5F 69084016 IC50 = 242 nM T69485 CKH1J6 69084057 IC50 = 410 nM T69485 C3WL1H 69084118 IC50 = 9 nM T69485 C4E9VH 69084152 IC50 = 217 nM T69485 CT2NK9 69084345 IC50 = 119 nM T69485 CQPA54 69084621 IC50 = 1080 nM T69485 C2P3LC 69085010 IC50 = 158 nM T69485 C4NU5T 69085032 IC50 = 106 nM T69485 C4SXT9 69085047 IC50 = 28 nM T69485 C8T0RS 69085151 IC50 = 3 nM T69485 C4RU6S 69085189 IC50 = 19 nM T69485 CA4U1J 69085230 IC50 = 35 nM T69485 C9WX0M 69085295 IC50 = 72 nM T69485 C4LM9J 69085642 IC50 = 29 nM T69485 CV76IC 69085689 IC50 = 395 nM T69485 C19PIM 69085726 IC50 = 43 nM T69485 C0Z1PN 69915149 Ki = 43 nM T69485 CP0N1Y 69915187 Ki = 15 nM T69485 C4I6UA 69915196 Ki = 5 nM T69485 C81MDP 69932186 Ki = 40 nM T69485 CA47RE 70169296 IC50 = 5 nM T69485 CHS9N3 70681618 IC50 < 1 nM T69485 CB2QP1 70681619 IC50 = 658 nM T69485 C4NVY5 70681620 IC50 = 96 nM T69485 CUS92R 70683739 IC50 = 23 nM T69485 CM41XZ 70683740 IC50 = 8 nM T69485 CAU6W8 70683741 IC50 = 8.7 nM T69485 CDL7J3 70683742 IC50 > 10000 nM T69485 C8PTI4 70685886 IC50 = 221 nM T69485 CWJ49Q 70685887 IC50 = 50 nM T69485 C5X8YM 70685888 IC50 = 447 nM T69485 C9O3RU 70685889 IC50 = 62 nM T69485 CFB9I0 70685890 IC50 < 1 nM T69485 CR7O0Q 70685891 IC50 = 2000 nM T69485 C8YIC1 70685892 IC50 = 7 nM T69485 C6B1TJ 70687123 IC50 = 170 nM T69485 C80BKR 70687129 IC50 = 220 nM T69485 C8G0AY 70688011 IC50 = 40 nM T69485 CTM9C1 70688012 IC50 = 13 nM T69485 C1IZ0S 70690040 IC50 = 4 nM T69485 CGA5E6 70690041 IC50 = 58 nM T69485 CCQR15 70690042 IC50 = 8 nM T69485 C3BRE9 70692193 IC50 = 2 nM T69485 CVT4S0 70692194 IC50 = 541 nM T69485 C0VL4I 70692195 IC50 = 137 nM T69485 C36FDI 70694255 IC50 = 82 nM T69485 CG4N1Z 70694256 IC50 = 151 nM T69485 CA58UO 70694257 IC50 = 125 nM T69485 C7UW0O 70696349 IC50 = 8 nM T69485 C0J2OK 70696350 IC50 = 40 nM T69485 CIPR26 70696351 IC50 = 2 nM T69485 CB3VS5 70816735 Ki > 2000 nM T69485 CWHM94 70816905 Ki = 108 nM T69485 C4RMS1 70817021 Ki = 949 nM T69485 C94LXI 70817051 Ki = 93 nM T69485 CSCO94 70817059 Ki = 1135 nM T69485 C7DO1N 70817239 Ki = 2 nM T69485 C6L7FH 70817382 Ki = 2 nM T69485 CTQ7C0 70818984 Ki = 367 nM T69485 CY03PE 70856594 Ki = 22 nM T69485 C7Q8ST 71522361 Ki = 1.1 nM T69485 C34TKD 71526207 Ki = 1.3 nM T69485 C2RO5Y 71526208 IC50 = 25 nM T69485 CZ7JD6 71527494 Ki = 0.1 nM T69485 C8NXQ0 71527606 Ki = 0.2 nM T69485 CE9SK3 71543409 Ki = 1.6 nM T69485 CR01NT 71555054 Ki = 9 nM T69485 CTS09B 71579478 IC50 = 111 nM T69485 C12KAY 71579479 IC50 = 13 nM T69485 CJN41M 71580771 IC50 = 194 nM T69485 C3QZ7D 71580772 IC50 = 24 nM T69485 CV8N1K 71580773 IC50 = 20 nM T69485 C4C9IF 71580858 IC50 = 225 nM T69485 CX6G8Z 71580859 IC50 = 2904 nM T69485 CW7K4I 71580860 IC50 = 29 nM T69485 CDC7T6 71580861 IC50 = 23 nM T69485 CQ2KC8 71580862 IC50 = 107 nM T69485 CL26RK 71580946 IC50 = 73 nM T69485 C9FIW3 71580947 IC50 = 2746 nM T69485 CAS05K 71580948 IC50 = 10 nM T69485 C0ND2T 71580949 IC50 = 194 nM T69485 C5WL4U 71580950 IC50 = 38 nM T69485 C1NL7J 71624633 Ki = 1.1 nM T69485 CWAY56 71716523 IC50 = 25 nM T69485 C1NP2M 72543760 IC50 = 11.6 nM T69485 CHU29Z 72699430 IC50 = 129 nM T69485 C1HMV0 72699854 IC50 = 2.73 nM T69485 CBF7O2 72699855 IC50 = 40.5 nM T69485 CKL84I 72699856 IC50 = 119 nM T69485 C1RY5X 72699949 IC50 = 23.6 nM T69485 C3I2OZ 72699950 IC50 = 2.57 nM T69485 CC70PO 72699951 IC50 = 139 nM T69485 C6HEI3 72700096 IC50 = 254 nM T69485 CH04OF 72700180 IC50 = 36 nM T69485 C5BKV3 72700181 IC50 = 532 nM T69485 CYJ2T4 72700265 IC50 = 80.1 nM T69485 CO7BI8 72700266 IC50 = 8.85 nM T69485 CL1U4W 72700267 IC50 = 61 nM T69485 CJN5K0 72700268 IC50 = 1310 nM T69485 CZ8K4T 72700362 IC50 = 471 nM T69485 C7BY8D 72700363 IC50 = 22.8 nM T69485 CHCM80 72700366 IC50 = 887 nM T69485 CZDM79 72700457 IC50 = 29 nM T69485 CTLC87 72700458 IC50 = 5.68 nM T69485 CSWL87 72700459 IC50 = 250 nM T69485 CPV92B 72700460 IC50 = 17.9 nM T69485 C5JT0D 72700462 IC50 = 11.3 nM T69485 CWZ0T6 72700543 IC50 = 5.87 nM T69485 CP8G5V 72700544 IC50 = 21.2 nM T69485 COSK78 72700626 IC50 = 1.61 nM T69485 C68GDU 72700698 IC50 = 43.2 nM T69485 CMP5F9 72703893 Ki = 309.03 nM T69485 C7ZAH6 72703894 Ki = 549.54 nM T69485 CW3NX0 72704097 Ki = 0.166 nM T69485 CEY4I0 72704098 Ki = 16.22 nM T69485 COTU10 72704099 Ki = 1.175 nM T69485 CGV76N 72704100 Ki = 4.571 nM T69485 CBE48L 72707143 Ki = 2.512 nM T69485 CO0U6I 72720554 Ki = 1.259 nM T69485 CVO7T2 72720555 Ki = 0.2512 nM T69485 CD8Z5T 72720556 Ki = 1.585 nM T69485 CXG47B 72720982 Ki = 0.631 nM T69485 CBW93F 72721081 Ki = 10 nM T69485 CHN0B5 72721178 Ki = 6.31 nM T69485 C4OD7F 72721280 Ki = 1 nM T69485 C41JEL 72721380 Ki = 0.7943 nM T69485 C50CDB 72721381 Ki = 6.31 nM T69485 CM45WC 72721691 Ki = 0.1995 nM T69485 CG8PX4 72721795 Ki = 1.995 nM T69485 CLD36Y 72721986 Ki = 1.585 nM T69485 C3JBG7 72721987 Ki = 0.5012 nM T69485 C82DJS 72722084 Ki = 0.1 nM T69485 CYC8U4 72722088 Ki = 5.012 nM T69485 C46UAR 72722089 Ki = 0.3981 nM T69485 C6Q3OM 72725148 Ki = 580 nM T69485 C3R1AC 72725149 Ki = 121 nM T69485 C8DAZ2 73346054 IC50 = 23 nM T69485 C2C7BU 73347449 IC50 = 9 nM T69485 CO7CY6 73347581 IC50 = 5 nM T69485 CB8F6U 73348981 IC50 = 10 nM T69485 C8KLQ1 73350080 EC50 = 850 nM T69485 CGZ7E4 73352057 IC50 = 16 nM T69485 CA9H1U 73353033 EC50 > 1000000 nM T69485 CJ4N5L 73353523 IC50 = 5 nM T69485 CB63NL 73356120 EC50 > 1000000 nM T69485 CIC73L 73356574 IC50 = 14 nM T69485 CH7S6O 73356708 Ki = 18 nM T69485 C15PYW 73673014 Ki = 0.5 nM T69485 C34LXD 74221626 Ki = 0.8 nM T69485 C6M7RX 74221720 Ki = 1.6 nM T69485 CN53AG 74221903 Ki = 2 nM T69485 CAIZ14 74221990 Ki = 5.1 nM T69485 C7SZG6 74222158 Ki = 0.4 nM T69485 C6J9LF 74222159 Ki = 3 nM T69485 C5J9EI 74222241 Ki = 1.3 nM T69485 CZA0I9 74222326 Ki = 0.7 nM T69485 C07NHS 74222327 Ki = 3.1 nM T69485 CGI5K2 74222402 Ki = 0.7 nM T69485 CZO3V4 74222406 Ki = 16.6 nM T69485 CL15XT 74222492 Ki = 3.4 nM T69485 CA1N8P 74222754 Ki = 8.9 nM T69485 CP9U0C 74222941 Ki = 2.6 nM T69485 CX5L0W 76072813 Ki = 0.9 nM T69485 CF5Z2M 76310080 Ki = 17 nM T69485 C28XZD 76310131 EC50 = 1610 nM T69485 CE5A0O 76310198 EC50 = 1360 nM T69485 CFS27O 76310208 EC50 = 263 nM T69485 CJO7X0 76310209 EC50 = 156 nM T69485 CE92OC 76310210 EC50 = 610 nM T69485 CG3RK5 76310211 EC50 = 1920 nM T69485 CLY90X 76310431 IC50 > 10000 nM T69485 C6W4YC 76310456 IC50 = 1070 nM T69485 CT20QS 76313798 EC50 = 1760 nM T69485 C9V7HM 76313820 EC50 = 99.3 nM T69485 C07WGU 76313901 EC50 = 3220 nM T69485 CF7J4U 76317345 EC50 = 1040 nM T69485 C5ZE9C 76317346 EC50 = 4820 nM T69485 CEVZ91 76317683 IC50 = 65 nM T69485 C6CFQ9 76321148 EC50 = 2180 nM T69485 CP8M6Z 76321165 EC50 = 2140 nM T69485 CM5HF7 76321386 IC50 = 771 nM T69485 C9DZN3 76324691 EC50 = 1250 nM T69485 C1XSG9 76324989 IC50 = 122 nM T69485 CB3K9C 76328274 EC50 = 3250 nM T69485 CR6W3T 76328275 EC50 = 729 nM T69485 C6I7AK 76328558 IC50 = 80 nM T69485 C3O9LC 76331924 EC50 = 439 nM T69485 CRUK21 76331925 EC50 = 1890 nM T69485 CVR8O9 76331964 EC50 = 1010 nM T69485 CC9AR4 76332010 EC50 = 1910 nM T69485 C54AVH 76332217 IC50 > 10000 nM T69485 C48LQC 76332218 IC50 = 416 nM T69485 CNK25I 76332219 IC50 = 1331 nM T69485 C0ZN3F 76332238 IC50 = 297 nM T69485 CA1Z7X 76335540 EC50 = 1990 nM T69485 CV8NM6 76335605 EC50 = 7850 nM T69485 CVK6J7 76335606 EC50 = 1440 nM T69485 CS2Y8O 76335607 EC50 = 2320 nM T69485 C2RVH7 76335608 EC50 = 1580 nM T69485 CRQ65T 76335879 IC50 > 10000 nM T69485 C0N3ZY 76534175 Ki = 10 nM T69485 CJG45W 76900605 Ki = 3.9 nM T69485 C81KEC 77105011 Ki > 1770 nM T69485 CNMG49 77105013 Ki > 2633 nM T69485 CZB61S 77105014 Ki > 4379 nM T69485 CI23UH 77105390 Ki > 2633 nM T69485 C45OVR 77106400 Ki = 4306 nM T69485 C91OPJ 77107393 Ki = 108 nM T69485 CLX8P9 77107592 Ki = 1227 nM T69485 CXS7B6 77107594 Ki = 521 nM T69485 CX0TB3 77107596 Ki = 379 nM T69485 CVK3R4 78324905 Ki = 1.3 nM T69485 CZ8FN7 86267288 IC50 = 2 nM T69485 CEQ2V4 86269345 IC50 = 0.7 nM T69485 C9WI2E 86271116 Ki = 221 nM T69485 C9PVK1 86276237 IC50 = 9 nM T69485 CF4QX9 86278359 Ki = 10 nM T69485 C0PUY4 86291876 Ki = 0.2 nM T69485 CK6WQ1 86291877 Ki = 0.4 nM T69485 CHB7U8 86291879 IC50 = 10 nM T69485 CR32FQ 86292273 Ki = 1.4 nM T69485 CU0NT8 86298249 Ki = 1.8 nM T69485 CH4XK1 86302551 Ki = 0.7 nM T69485 CL7C5E 86302552 Ki = 9.2 nM T69485 C47MVU 86695644 IC50 = 20 nM T69485 CK9I5Y 89789751 IC50 = 2 nM T69485 C39TXO 89789760 IC50 = 5 nM T69485 C9I6NQ 89789762 IC50 = 3 nM T69485 C8S7BC 89789778 IC50 = 2 nM T69485 C0M7SQ 89789795 IC50 = 5 nM T69485 CERC67 89789843 IC50 = 4 nM T69485 CC1XN6 90286209 Ki = 1137 nM T69485 CSJ05B 90286221 Ki = 467 nM T69485 CQ1DK9 90286288 Ki = 220 nM T69485 CZU57Y 90286316 Ki = 1564 nM T69485 C2V5TA 90286327 Ki = 521 nM T69485 CWP4H0 90286502 Ki = 467 nM T69485 CQE2R4 90298269 Ki = 627 nM T69485 C81IGW 90298273 Ki = 193 nM T69485 C42HYM 90298275 Ki = 2143 nM T69485 C1TU7S 90298326 Ki > 1935 nM T69485 C3FD8G 90298333 Ki > 2096 nM T69485 C5OYE8 90298382 Ki = 933 nM T69485 CZ6X9P 90298385 Ki = 1470 nM T69485 CT7C1S 90298426 Ki = 271 nM T69485 C81JWB 90298427 Ki = 1409 nM T69485 CAO2H3 90298431 Ki = 120 nM T69485 CY9O3G 90405964 Ki = 562 nM T69485 C2WGJ3 90654337 Ki = 25 nM T69485 C8YE0S 90654338 Ki = 0.53 nM T69485 CZIE39 90654339 Ki = 26 nM T69485 C6TGU4 90654340 Ki = 3 nM T69485 CK38IX 90654341 Ki = 28 nM T69485 CL7KM1 90654342 Ki = 11 nM T69485 CFQS07 90654343 IC50 = 28 nM T69485 C8APK1 90654344 Ki = 7 nM T69485 C71YVR 90654345 Ki = 24 nM T69485 C2E5MT 90654346 Ki = 7.5 nM T69485 CPKH23 90654347 Ki = 130 nM T69485 CN7CX5 90654348 Ki = 5.6 nM T69485 CF0T9O 90654349 Ki = 42 nM T69485 C37MYP 90654350 Ki = 150 nM T69485 CJT36M 90654351 Ki = 32 nM T69485 CJ0Z5H 90656176 Ki = 1.5 nM T69485 CCW7S2 90656177 Ki = 0.3 nM T69485 C3EN1D 90656178 Ki = 49 nM T69485 CRK0W5 90656179 Ki = 92 nM T69485 CDN8Y4 90656180 Ki = 5 nM T69485 CJUS40 90656181 Ki = 25 nM T69485 CPSI06 90656182 Ki = 0.4 nM T69485 C8ZFG3 91801202 Ki = 1.259 nM T69485 C0DFT8 91809243 Ki = 2.6 nM T69485 CP0CE9 91810287 EC50 = 23 nM T69485 CXO4N6 117668910 Ki = 3.9 nM T69485 C4HZ0N 117857721 IC50 = 13.5 nM T69485 CJA8G5 117859490 IC50 = 14 nM T69485 C1O2AH 117859572 IC50 = 19 nM T69485 C0CPN6 117859931 IC50 = 14 nM T69485 CZ20RX 118020300 IC50 = 58.4 nM T69485 C2Z1IN 118020504 IC50 = 952 nM T69485 CNI86H 118020539 IC50 = 840 nM T69485 CNKV57 118167452 Ki = 1.7 nM T69485 CSA7U9 118175269 Ki = 2.2 nM T69485 C72NVT 118175279 Ki = 0.8 nM T69485 CDAS04 118180165 Ki = 0.4 nM T69485 CK90HX 118435993 Ki = 1.7 nM T69485 C71DSJ 118496811 Ki = 871 nM T69485 CU45VI 118504517 Ki > 3327 nM T69485 CF52MN 118715605 Ki = 43 nM T69485 C4VR8L 118715606 Ki = 11 nM T69485 CG8MX4 118715607 Ki = 11 nM T69485 C1WKZ9 118715608 Ki = 140 nM T69485 CW4Z5M 118715609 Ki = 1.4 nM T69485 CN36LS 118715610 Ki = 193 nM T69485 C51JPK 118715611 Ki = 5.2 nM T69485 C1J2CY 118715612 Ki = 75 nM T69485 CN14EP 118715613 Ki = 4.1 nM T69485 CNWA97 118716929 Ki = 8654 nM T69485 C3NW1S 118716930 Ki > 10000 nM T69485 CI3TK2 118716931 Ki = 4226 nM T69485 C5WRI1 118716932 Ki = 7.2 nM T69485 C5OQ4Y 118716933 Ki = 7846 nM T69485 C36PCB 118716934 Ki = 4679 nM T69485 CCT4Y0 118716935 Ki > 10000 nM T69485 CWJ69M 118716936 Ki = 967 nM T69485 C9YEL0 118716937 Ki = 129 nM T69485 CG5R1B 118716938 Ki = 588 nM T69485 CHK4C7 118716939 Ki = 1330 nM T69485 CG75OB 118716940 Ki = 384 nM T69485 CG52QK 118716941 Ki = 3336 nM T69485 C0QS6Y 118716942 Ki = 51 nM T69485 C10SEV 118716943 Ki = 85 nM T69485 CAF89K 118716944 Ki = 35 nM T69485 C60JTD 118716945 Ki = 14 nM T69485 C2U1BX 118716946 Ki = 28 nM T69485 C83SPX 118716947 Ki = 27 nM T69485 C5ELB1 118716948 Ki = 34 nM T69485 C37UXI 118726303 Ki = 8.9 nM T69485 CFN4Y7 118726304 Ki = 55 nM T69485 C1Z7TR 118726305 Ki = 18 nM T69485 CX51TS 118726306 Ki = 1 nM T69485 C68ITL 118726307 Ki = 149 nM T69485 C62FYU 118726308 Ki = 180 nM T69485 CLQ34R 118726309 Ki = 5.2 nM T69485 CZ3OB5 118726310 Ki = 2.6 nM T69485 C9WN2G 118726311 Ki = 0.9 nM T69485 CHM76O 118726312 Ki = 63 nM T69485 C5S4RU 118726313 Ki = 1.1 nM T69485 CS09EU 118726314 Ki = 0.8 nM T69485 C43OAN 118726315 Ki = 370 nM T69485 CN2KE3 118731950 IC50 > 10000 nM T69485 CF4QD0 118731951 IC50 = 9490 nM T69485 CYNB60 118731952 IC50 = 2050 nM T69485 C0VU1B 118731953 IC50 > 10000 nM T69485 CH8T0S 118731954 IC50 = 5810 nM T69485 C7KX2R 118731955 IC50 = 8300 nM T69485 CWA05F 118731956 IC50 > 10000 nM T69485 CC3PT6 118731957 IC50 = 5 nM T69485 CXEO47 118731958 IC50 = 315 nM T69485 CTY98B 118736949 Ki = 7.6 nM T69485 C19HQW 118736950 Ki = 2.6 nM T69485 CRJ9L8 118736951 Ki = 2400 nM T69485 C82NQB 118736952 Ki = 0.6 nM T69485 CVO72M 118736953 Ki = 0.6 nM T69485 CWH08B 118736954 Ki = 6.5 nM T69485 CLAR49 118736955 Ki = 0.2 nM T69485 C3G6VD 118736956 Ki = 0.9 nM T69485 CCK3A9 118736957 Ki = 4.5 nM T69485 CYBN01 118736958 Ki = 3.8 nM T69485 CLNY63 118736959 IC50 = 21 nM T69485 CNU4D7 118736960 IC50 = 21 nM T69485 CKFZ15 118736961 IC50 = 38 nM T69485 COPD90 118736962 IC50 = 37 nM T69485 CJ3VD1 118736963 IC50 = 32 nM T69485 CMRB20 121231398 Ki = 4.5 nM T69485 CYHP86 122179999 Ki > 2000 nM T69485 CI3Q9N 122180000 Ki = 204 nM T69485 CND0S5 122180001 Ki = 8 nM T69485 C0T3SD 122180002 Ki = 49 nM T69485 C6CG5E 122180317 Ki = 1600 nM T69485 CQR14H 122180318 Ki = 510 nM T69485 CE36GC 122180319 Ki = 680 nM T69485 CVL0Q7 122180320 Ki = 875 nM T69485 CW8H2J 122180321 Ki = 746 nM T69485 CS1JC7 122180322 Ki = 687 nM T69485 C6FVZ0 122180323 Ki = 294 nM T69485 CX9JG0 122180324 Ki = 137 nM T69485 CQU2H9 122180325 Ki = 421 nM T69485 CA5CP8 122180326 Ki = 240 nM T69485 C6CAZ0 122180327 Ki = 899 nM T69485 CRVB56 122180328 Ki = 768 nM T69485 CAL3T2 122180329 Ki = 106 nM T69485 C3OJS0 122180330 Ki = 9.8 nM T69485 C4YIX5 122180331 Ki = 51 nM T69485 C2DZ3Y 122180332 Ki = 141 nM T69485 C0W3JG 122180333 Ki = 180 nM T69485 C6EF1H 122180334 Ki = 27 nM T69485 C8SD7F 122180335 Ki = 41 nM T69485 C2WV9G 122180336 Ki = 12 nM T69485 CJ1AP3 122180337 Ki = 14 nM T69485 CBN0J2 122180338 Ki = 10 nM T69485 CEA80S 122180339 Ki = 30 nM T69485 CTG4B2 122180340 Ki = 30 nM T69485 C6Y0JD 122180341 Ki = 120 nM T69485 CTCN25 122180342 Ki = 54 nM T69485 C35BFD 122180343 Ki = 8 nM T69485 C80QZN 122180344 Ki = 46 nM T69485 C6YIR4 122180345 Ki = 77 nM T69485 CO1AK6 122184039 Ki = 1 nM T69485 C5XOD3 122184040 Ki = 44 nM T69485 CAYV10 122184041 IC50 = 6 nM T69485 CUWG52 122184042 Ki = 571 nM T69485 CTL34Z 122184043 Ki = 12 nM T69485 CVRO25 122184044 Ki = 800 nM T69485 C3WUY1 122184045 Ki = 189 nM T69485 CCG80F 122191738 Ki = 3600 nM T69485 C65BVD 122191739 Ki = 850 nM T69485 CKOL57 122191740 Ki = 1800 nM T69485 C8XA6F 122191741 Ki = 6.1 nM T69485 CSR2P0 122191742 Ki = 3.9 nM T69485 CH20JU 122191743 Ki = 14 nM T69485 CG23UT 122191744 Ki = 5.1 nM T69485 C1IOQ4 122191745 Ki = 1100 nM T69485 CGOL70 122191746 Ki = 4200 nM T69485 CM1KR0 122191747 Ki = 760 nM T69485 CJKH54 122191748 IC50 = 245 nM T69485 CF74NG 122191819 EC50 > 10000 nM T69485 COY58Z 122191820 EC50 = 800 nM T69485 CNK5E4 122191821 EC50 > 10000 nM T69485 CW4P2C 122191822 EC50 = 182 nM T69485 C9HF4M 122191823 EC50 = 50 nM T69485 CB4VN2 122191824 EC50 = 235 nM T69485 CQC31A 122191825 EC50 > 1000 nM T69485 CV47JA 122191826 EC50 > 10000 nM T69485 C9PTF1 122191827 EC50 = 268 nM T69485 CX4WR3 122191828 EC50 > 10000 nM T69485 CBI0X1 122191829 EC50 = 33 nM T69485 C7VA3T 122191830 EC50 = 1047 nM T69485 CW7F8P 122192246 EC50 = 800 nM T69485 CQ8FE7 122192247 EC50 = 31 nM T69485 C5YRQ9 122192248 EC50 = 94 nM T69485 CMX26J 122192250 EC50 = 28 nM T69485 C4TX5S 122195752 Ki = 10 nM T69485 CKE37J 123517068 Ki = 1617 nM T69485 CD57NR 127027859 Ki = 22 nM T69485 CM91FC 127037650 IC50 = 3.5 nM T69485 CBT18A 127037651 IC50 = 65 nM T69485 CLD41N 127037996 IC50 = 3.3 nM T69485 C8INE9 127038060 IC50 = 4.7 nM T69485 CC3T8J 127038061 IC50 = 4 nM T69485 CJ03FI 127038062 IC50 = 3.1 nM T69485 CACI97 127038343 IC50 = 71 nM T69485 C4P7YM 127038416 IC50 = 12 nM T69485 C54FRL 127038812 IC50 = 40 nM T69485 CV6QR8 127038813 IC50 = 4.3 nM T69485 CRE04H 127038817 IC50 = 10 nM T69485 C71SOB 127038818 IC50 = 66 nM T69485 CRY01S 127038819 IC50 = 62 nM T69485 CSHM50 127038820 IC50 = 6.3 nM T69485 CNG1V0 127038821 IC50 = 6.6 nM T69485 CW47SG 127038822 IC50 = 8 nM T69485 CV8Z7T 127039127 IC50 = 1.8 nM T69485 CVOW03 127039128 IC50 = 16 nM T69485 C5IX1B 127039129 IC50 = 18 nM T69485 C1YUH6 127039134 IC50 = 7.8 nM T69485 C1NZ6H 127039135 IC50 = 10 nM T69485 CIBD78 127040414 IC50 = 102 nM T69485 COM28D 127040734 IC50 = 428 nM T69485 C37QEO 127040735 IC50 = 16 nM T69485 C6DEH8 127040736 IC50 = 243 nM T69485 CAX2I9 127040737 IC50 = 8.4 nM T69485 CTW7A2 127041999 Ki = 63.1 nM T69485 C07JPS 127042658 IC50 = 39 nM T69485 CDG71E 134132166 Ki > 5868 nM T69485 CE3G0J 134134612 Ki = 861 nM T69485 CTU5I2 134136264 Ki = 18 nM T69485 C76TDR 134137910 Ki > 12660 nM T69485 CC76IK 134139865 Ki = 281 nM T69485 CSTW95 134141417 Ki = 11 nM T69485 CPR6S3 134142016 Ki = 277 nM T69485 C5X7JG 134142573 Ki = 2.8 nM T69485 CFH62V 134143971 Ki > 3370 nM T69485 CD2H4Y 134144793 Ki = 9 nM T69485 C5P1YI 134144954 Ki = 1009 nM T69485 C8Q5WK 134150272 Ki = 1038 nM T69485 C4YS1O 134150303 Ki > 12720 nM T69485 CDR51U 134151486 Ki > 1407 nM T69485 C5UFJ1 134151826 Ki > 4379 nM T69485 CP1V5L 134152443 Ki = 907 nM T69485 CFP4Q5 134153918 Ki = 27 nM T69485 C0ZAO5 134155036 Ki > 4379 nM T69485 CM87PX 134155753 Ki = 14 nM T69485 CU58RD 135314438 Ki > 10000 nM T69485 CPZ89B 135314564 Ki > 10000 nM T69485 C24MIN 137632538 IC50 = 1269 nM T69485 C3UBF8 137634720 IC50 = 238 nM T69485 C0BRG6 137636340 IC50 = 211 nM T69485 C0G8TB 137637342 IC50 = 1822 nM T69485 C7FUO1 137638475 Ki > 10000 nM T69485 C04EGF 137638805 IC50 = 131 nM T69485 CYB93R 137638895 IC50 = 1044 nM T69485 CZ91SV 137638898 IC50 > 10000 nM T69485 CT90FM 137640166 IC50 = 4845 nM T69485 CIPJ41 137641369 IC50 = 791 nM T69485 C5OXI1 137642484 IC50 = 639 nM T69485 CX3MK7 137642825 IC50 = 5988 nM T69485 C2DIV4 137644135 IC50 >= 10000 nM T69485 C6M0BL 137644509 IC50 = 108 nM T69485 C9ABK7 137644534 IC50 = 1185 nM T69485 C2MRK0 137645329 Ki = 2070 nM T69485 C9GP2E 137645716 Ki = 0.7 nM T69485 CC6KI7 137646689 IC50 = 4710 nM T69485 CF98UE 137647371 IC50 = 1524 nM T69485 C2BQ4U 137648163 IC50 = 2787 nM T69485 C4VD0P 137649196 IC50 > 10000 nM T69485 CLZ2N8 137649834 IC50 = 206 nM T69485 C1TW0K 137650367 Ki = 0.6 nM T69485 C7X0SU 137651169 IC50 > 10000 nM T69485 CR5F0I 137652411 IC50 = 178 nM T69485 C08XSJ 137655492 IC50 > 10000 nM T69485 C1MJG9 137655850 IC50 = 775 nM T69485 C7R3IU 137656102 Ki = 725 nM T69485 CQ0UG7 137657078 IC50 = 354 nM T69485 C7VFU4 137657849 IC50 = 1093 nM T69485 CF7Q6D 137658206 IC50 = 575 nM T69485 C63RQO 137658775 IC50 = 387 nM T69485 C89FIO 137659457 IC50 = 508 nM T69485 CNH3U0 137660075 IC50 = 1685 nM T69485 C38LZW 137660448 Ki = 294 nM T69485 CQ0J2X 137660887 IC50 = 311 nM T69485 CUMN86 137662108 Ki = 2.5 nM T69485 CZ4S3O 144671360 IC50 > 5868 nM T69485 CF0Z8D 145714283 Ki = 50.12 nM T69485 CS9B7W 145971593 Ki > 10000 nM T69485 C27YQH 145975735 Ki > 10000 nM T69485 C7CO2P 145977763 Ki = 123 nM T69485 C6VWK3 145979924 Ki = 3600 nM T69485 CGRU50 145989367 Ki = 4300 nM T69485 C3M1WQ 145994245 Ki = 3200 nM T69485 CHIZ91 153284501 IC50 = 2260 nM T69485 CQD73L 155515631 Ki > 10000 nM T69485 C2B1ZG 155517489 Ki > 10 nM T69485 CH3MT0 155519961 Ki > 10 nM T69485 C9D3AS 155520434 Ki > 10000 nM T69485 CF1N4P 155524300 Ki > 10000 nM T69485 CWL04C 155524427 Ki = 79.9 nM T69485 CB3JY5 155525887 Ki > 10000 nM T69485 C5EM4D 155532688 Ki = 173 nM T69485 C4VQ8A 155543013 Ki > 10 nM T69485 CP7I4W 155543165 Ki > 10 nM T69485 CFMK42 155543728 Ki > 10 nM T69485 CIY9N3 155554119 Ki > 10 nM T69485 CQ30PW 155557825 Ki > 10 nM T69485 CRDS43 155566853 Ki > 10 nM T69485 CM93SV 155567436 Ki = 91.9 nM T69485 CQ1RW5 155568320 Ki > 10000 nM T69485 D01SUL 9869934 Ki = 5.012 nM T69485 D02MDC 9981404 Ki = 1.1 nM T69485 D08MXD 73349109 Ki = 129 nM T69485 D0J3PJ 4331799 Ki = 794.33 nM T69485 D0KP3K 10065953 Ki = 503 nM T69485 D0R4BT 10046856 Ki = 100 nM T69485 D0U0TS 10408514 IC50 = 40 nM T69485 D0UZ4J 6604926 Ki = 630.96 nM T95923 C4Z7TA 128167 Ki = 39 nM T95923 C2MU3S 753410 Ki = 1084 nM T95923 CPA98T 869604 IC50 = 4504 nM T95923 C4ESQ9 1105689 Ki = 7020 nM T95923 CYQ7L5 1365686 Ki = 230 nM T95923 CRD4O3 2230607 Ki = 316.6 nM T95923 C4TGR0 2260227 Ki = 310 nM T95923 C32MJD 3114900 IC50 = 6600 nM T95923 CN8XM2 5311263 EC50 = 77 nM T95923 CWIH09 5311306 IC50 = 6450 nM T95923 CO15VM 5353734 EC50 ~ 10 nM T95923 CAX9U1 5473680 EC50 > 11800 nM T95923 CDM1E9 5861754 IC50 = 30 nM T95923 CLS96Y 6419701 EC50 = 575.44 nM T95923 C9R7UG 6610239 EC50 = 1600 nM T95923 CA78VE 9958483 IC50 = 40 nM T95923 C9EQ7R 9960370 IC50 = 6450 nM T95923 C8IGL1 10136738 EC50 > 5000 nM T95923 COZF72 10322404 EC50 = 0.2692 nM T95923 CE1Y9O 10393842 IC50 = 175 nM T95923 C5CQ0S 10410675 EC50 = 683.7 nM T95923 CPS0Z3 10432221 EC50 = 112.6 nM T95923 C6ABN7 10927764 EC50 > 10000 nM T95923 CO1N7Q 11015922 EC50 > 10000 nM T95923 C9EDZ5 11026029 EC50 ~ 3000 nM T95923 C1MRI2 11080129 EC50 > 10000 nM T95923 CLJ0N4 11101949 Ki = 119 nM T95923 COID45 11122865 EC50 > 10000 nM T95923 CB94ZA 11178884 EC50 ~ 500000 nM T95923 CIF3K9 11312936 Ki = 76 nM T95923 CQLP42 11473989 EC50 = 546 nM T95923 CRCF96 11512311 IC50 > 10000 nM T95923 CFHV74 11568387 Ki = 5 nM T95923 C2JDN7 11592067 IC50 > 10000 nM T95923 CIZW04 11599847 IC50 = 642 nM T95923 C0CBY2 11625765 EC50 = 3 nM T95923 C7QRT8 11648176 EC50 = 0.2239 nM T95923 CAW3R6 11732670 EC50 > 10000 nM T95923 CY3L7V 11755685 Ki = 2325 nM T95923 CK7O0X 11849496 Ki = 1150 nM T95923 CV2HM3 12109913 EC50 ~ 1000 nM T95923 CG80FP 12109914 EC50 > 10000 nM T95923 CYL31W 12109920 EC50 ~ 20000 nM T95923 CR79CQ 16043259 Ki = 636 nM T95923 CZO6H5 16045222 EC50 = 115 nM T95923 CZ1C9V 23629653 IC50 = 143 nM T95923 C70ONJ 23725184 Ki = 512 nM T95923 C1F9GI 24882686 IC50 > 50000 nM T95923 CR2M4K 44325214 IC50 > 10000 nM T95923 C6KE2Z 44325235 IC50 > 10000 nM T95923 C15FHI 44325304 IC50 > 10000 nM T95923 CW3XH1 44325312 IC50 > 10000 nM T95923 CI2YX1 44325339 IC50 > 10000 nM T95923 C9ZNP8 44325351 IC50 = 6930 nM T95923 CT82OZ 44325364 IC50 = 5920 nM T95923 CS0A5D 44325365 IC50 = 351 nM T95923 COS7A5 44325366 IC50 = 3280 nM T95923 CT0RI4 44325370 IC50 = 6410 nM T95923 C16ENI 44325390 IC50 = 4030 nM T95923 CL6Q4T 44325391 IC50 = 35.6 nM T95923 C8O6ZB 44325400 IC50 = 427 nM T95923 CE1QC6 44325401 IC50 = 2310 nM T95923 C19LDV 44325402 IC50 > 10000 nM T95923 CG5N0T 44325416 IC50 > 10000 nM T95923 CD4AI9 44325421 IC50 = 6840 nM T95923 CDQ8P0 44325422 IC50 = 7220 nM T95923 CJI36T 44325680 IC50 = 9260 nM T95923 C2VWE0 44325681 IC50 = 2630 nM T95923 CMEB29 44325682 Ki = 940 nM T95923 C4F8UE 44343851 EC50 > 5000 nM T95923 CD1SX3 44343866 EC50 > 5000 nM T95923 CK0NG4 44343867 EC50 > 5000 nM T95923 C5J4BE 44343880 EC50 > 5000 nM T95923 CS7BJ1 44344023 EC50 > 5000 nM T95923 CV86RF 44368508 EC50 = 0.44 nM T95923 CD6ZL8 44392725 Ki = 1156 nM T95923 CV80NT 44392726 Ki = 2600 nM T95923 CSQ0E4 44392727 Ki > 10000 nM T95923 C0U3XC 44392738 Ki > 10000 nM T95923 CHA7T6 44392762 Ki = 6236 nM T95923 CP8S6X 44392769 Ki = 2075 nM T95923 CTKZ61 44392778 Ki = 6960 nM T95923 CNVU84 44392779 Ki = 455 nM T95923 CXL4U0 44392780 Ki = 1093 nM T95923 CUH71K 44392791 Ki = 102 nM T95923 C4Y8HZ 44392792 Ki = 39 nM T95923 CTNU76 44392793 Ki = 48 nM T95923 CM3RG9 44392794 Ki = 1660 nM T95923 C1Y8ME 44392795 Ki = 423 nM T95923 CCOF81 44392796 Ki = 39 nM T95923 CKF5A4 44392797 Ki = 561 nM T95923 CGPA21 44392798 Ki = 533 nM T95923 CUR57A 44392834 Ki = 1050 nM T95923 CR17IB 44392835 Ki = 150 nM T95923 CBR7Y6 44392836 Ki = 4000 nM T95923 C6T1DR 44394293 Ki = 196 nM T95923 CJUO17 44397968 Ki = 588 nM T95923 C6KWD8 44400304 EC50 ~ 10 nM T95923 CAE68N 44400338 EC50 > 10000 nM T95923 C6GM3O 44400339 EC50 ~ 5000 nM T95923 C05VIO 44400351 EC50 > 10000 nM T95923 C8BNL6 44400365 EC50 ~ 200 nM T95923 C7MDS6 44400374 EC50 > 10000 nM T95923 CI7CM0 44400377 EC50 > 10000 nM T95923 CGEY06 44400378 EC50 ~ 5000 nM T95923 CPW4T1 44400380 EC50 ~ 1000 nM T95923 C5IM9X 44400388 EC50 ~ 500 nM T95923 C8YKT7 44400424 EC50 ~ 10000 nM T95923 C38LAH 44400430 EC50 ~ 500000 nM T95923 C9ISN4 44407385 Ki = 489 nM T95923 C5LAU4 44407386 Ki = 117 nM T95923 C9P3SU 44407394 Ki = 50 nM T95923 C9E2RP 44407397 EC50 = 164 nM T95923 CWN45J 44407485 Ki = 118 nM T95923 C8OB1A 44414925 Ki = 3170 nM T95923 C3SX2V 44414935 EC50 > 7030 nM T95923 C29TWV 44454059 IC50 > 50000 nM T95923 CO7L3S 44454369 IC50 = 12000 nM T95923 CY7ZA1 44586491 IC50 = 184 nM T95923 C85ANH 46213949 IC50 > 8000 nM T95923 CET63X 46223906 EC50 = 0.2754 nM T95923 C8CK4M 46240292 IC50 = 1600 nM T95923 C95UCQ 58787991 EC50 = 321.8 nM T95923 CNM5Y7 66553162 IC50 = 8340 nM T95923 C9GQ2D 66774612 IC50 > 10000 nM T95923 CW2O5R 66774777 IC50 > 10000 nM T95923 CKL76D 66775043 IC50 > 10000 nM T95923 C9NYD7 70819486 IC50 > 30000 nM T95923 C7GFM8 70819507 IC50 > 30000 nM T95923 CN13BI 70856266 IC50 = 2290 nM T95923 C19LCA 71264582 IC50 > 500 nM T95923 CFY03B 71450323 IC50 > 30000 nM T95923 CR6LV5 71452129 IC50 = 2310 nM T95923 C8BJ1R 71452130 IC50 = 5800 nM T95923 CLZI05 71452131 IC50 = 8260 nM T95923 CET67P 71453960 IC50 = 21940 nM T95923 CJ4ZR7 71453961 IC50 > 30000 nM T95923 C2YZP4 71455702 IC50 = 6860 nM T95923 C43TXF 71455703 IC50 = 27350 nM T95923 C80YTO 71455704 IC50 = 6300 nM T95923 CQMU34 71457480 IC50 = 132 nM T95923 CZH0Q5 71457481 IC50 = 65 nM T95923 CI4T3M 71457482 IC50 = 18600 nM T95923 C2YO9B 71457483 IC50 > 30000 nM T95923 CG0ZL8 71461122 IC50 > 30000 nM T95923 C2MPI8 71461123 IC50 > 30000 nM T95923 C4NU2T 71461124 IC50 > 30000 nM T95923 CID7N8 71461125 IC50 > 30000 nM T95923 C4QTR2 71462858 IC50 = 478 nM T95923 C06NYA 71462863 IC50 > 30000 nM T95923 C57TYK 71569053 EC50 = 0.36 nM T95923 CSN3I7 71569056 EC50 = 0.2042 nM T95923 CPT5S2 71718248 EC50 = 0.39 nM T95923 CKC4U7 71719457 EC50 = 1.072 nM T95923 C5P1CQ 71720690 EC50 = 0.37 nM T95923 CX71VH 73348672 IC50 = 24 nM T95923 CQ6B3X 90665720 Ki = 48 nM T95923 CG65XZ 122191108 Ki = 170 nM T95923 CQ3W8I 122191543 EC50 = 62 nM T95923 CWQ8Y3 122191544 IC50 = 1160 nM T95923 CO5Y0B 122191545 IC50 = 2300 nM T95923 D02LXI 10367662 Ki = 148 nM T95923 D02RYR 11447695 Ki = 504 nM T95923 D03HLU 11276402 Ki = 370 nM T95923 D04BLL 11312382 Ki = 40 nM T95923 D04CJG 82327 Ki = 211 nM T95923 D04KQT 10468943 Ki = 14 nM T95923 D05TVG 23682233 Ki = 170 nM T95923 D06YTN 81309 Ki = 680 nM T95923 D07WLV 11219269 Ki = 27 nM T95923 D07YUV 11197104 Ki = 58 nM T95923 D0BP3E 11393306 Ki = 575 nM T95923 D0D5OY 44400349 EC50 ~ 20000 nM T95923 D0E0DY 62532 Ki = 121 nM T95923 D0F2SQ 11288209 Ki = 128 nM T95923 D0G6XT 10051843 Ki = 202 nM T95923 D0GH9J 44407389 Ki = 67 nM T95923 D0H6DZ 16078994 EC50 = 276 nM T95923 D0N4AG 11220562 Ki = 14 nM T95923 D0P7GR 78401 Ki = 1120 nM T95923 D0PI4H 10282223 IC50 > 10000 nM T95923 D0R8LB 44343825 EC50 > 5000 nM T95923 D0S6CW 44392752 Ki = 1688 nM T95923 D0U5US 78816 Ki = 303 nM T95923 D0X0OP 56947064 EC50 = 80 nM T95923 D0X0UR 5497152 EC50 = 290 nM T95923 D0XJ9P 75816 Ki = 121 nM T95923 D0XY0Z 11208266 Ki = 14 nM T95923 D0Z2QV 11242245 Ki = 49 nM T25462 CBX8T9 16451230 IC50 > 150000 nM T25462 C52WPZ 53356803 Ki < 1 nM T25462 C5JOC6 54766612 Ki < 1 nM T25462 CBT35C 54766613 Ki < 1 nM T25462 C8IPK7 71586081 IC50 = 320 nM T25462 CDP4G0 72710747 IC50 = 800 nM T25462 C4XJ5N 78357767 IC50 > 100000 nM T25462 D02TVQ 71268957 IC50 > 100000 nM T25462 D09CLP 439155 IC50 = 2300 nM T58496 D0CO6D 71144018 IC50 > 20000 nM T58496 COL7M1 17421069 IC50 > 20000 nM T58496 C7FBO1 25270198 IC50 > 100000 nM T58496 C23WVS 53361524 IC50 > 10000 nM T58496 CBF0S5 56652700 IC50 = 160 nM T58496 C8WVE2 71554840 IC50 = 380 nM T58496 CN61RW 90645447 IC50 > 30000 nM T58496 CISP03 90645459 IC50 > 30000 nM T58496 CM5FN9 90645460 IC50 > 30000 nM T58496 C31TXQ 90645465 IC50 > 30000 nM T58496 C6OF3B 90645468 IC50 > 30000 nM T58496 C0VW1K 90645470 IC50 > 30000 nM T58496 C1XNR3 121513880 IC50 > 30000 nM T58496 D0D6MC 1150897 IC50 > 10000 nM T22658 D09BHB 5509 IC50 = 90 nM T22658 D0R1RS 3715 IC50 = 50 nM T22658 D0TG1H 3033 IC50 = 8 nM T22658 D0ZL4F 180540 IC50 = 20 nM T22658 CCZ3K9 15250 IC50 > 1000 nM T22658 C4PG1B 30931 IC50 > 1000 nM T22658 CNB6V7 114864 IC50 = 50 nM T22658 C7AKH8 141222 IC50 > 1000 nM T22658 C6EVL8 854057 IC50 > 1000 nM T22658 CNRE12 13309832 IC50 > 1000 nM T22658 CRB2H6 14762946 IC50 = 500 nM T22658 CNJ72V 18546323 IC50 > 1000 nM T22658 C5FD2Z 22218600 IC50 > 1000 nM T22658 CM3NT2 44298341 Ki = 13000 nM T22658 CX79VC 45268160 IC50 > 1000 nM T22658 C95IAE 45269044 IC50 = 600 nM T22658 CS2JM1 45269050 IC50 = 12 nM T22658 CEGP42 45269893 IC50 = 50 nM T22658 C5TE3O 45269894 IC50 = 13 nM T22658 C4O9EY 45269895 IC50 = 650 nM T22658 C34QNT 45269905 IC50 = 10 nM T22658 CGVT73 45270722 IC50 = 20 nM T22658 C4KH1C 45272452 IC50 = 25 nM T22658 C03KDJ 78224453 Ki = 7000 nM T22658 C0M8ZV 134130686 Ki = 106000 nM T22658 C1AS4F 134130687 Ki = 4000 nM T22658 CG0QB1 134130688 Ki = 12000 nM T22658 CFZG03 134130848 Ki = 10000 nM T22658 CGH9T1 134130849 Ki = 13000 nM T22658 CGW47R 134130850 Ki = 14000 nM T22658 C1NY6S 134130851 Ki = 6000 nM T22658 C2B3KN 134130852 Ki = 31000 nM T22658 CA0X3S 134130853 Ki = 4000 nM T22658 C42SCP 134130854 Ki = 383000 nM T22658 CD1TK0 134130855 Ki = 9300 nM T22658 CG35UE 134130856 Ki = 2300 nM T22658 D05EMX 14076674 IC50 = 25 nM T22658 D08GOT 13752584 IC50 = 400 nM T22658 D0I8YN 18546352 IC50 = 9 nM T22658 D0Q8ZV 15581854 IC50 = 500 nM T22658 D0T8RL 13409348 IC50 = 13 nM T50914 CC7KZ4 8902460 IC50 = 23000 nM T50914 CM4IH2 16353955 IC50 < 20000 nM T50914 CQ2G5U 17456976 IC50 < 20000 nM T50914 C2X8LS 17456979 IC50 < 20000 nM T50914 C25WOJ 24450633 IC50 < 20000 nM T50914 CKB35V 31263096 IC50 < 20000 nM T50914 CI25OW 31264587 IC50 < 20000 nM T50914 CTPQ58 45280035 IC50 = 480 nM T50914 CI1QN6 70983932 IC50 = 86.3 nM T50914 CNO40E 73387017 IC50 > 100000 nM T50914 CQ10IZ 73387018 IC50 < 20000 nM T50914 CM6E5I 73387106 IC50 < 20000 nM T50914 C4RCS2 73387109 IC50 < 20000 nM T50914 CI4TM7 73387207 IC50 < 20000 nM T50914 C15RGZ 73387208 IC50 < 20000 nM T50914 CJKE78 73387209 IC50 < 20000 nM T50914 C7A4LV 73387210 IC50 < 20000 nM T50914 CHU7M4 73387294 IC50 < 20000 nM T50914 CDJS39 73387295 IC50 < 20000 nM T50914 C87XME 73387296 IC50 < 20000 nM T50914 CAQ63J 73387298 IC50 < 20000 nM T50914 CM93DI 76332066 Ki = 150 nM T50914 C8C7JV 118707614 IC50 < 20000 nM T50914 C23ALW 118707615 IC50 < 20000 nM T50914 CDF7R4 118707616 IC50 < 20000 nM T50914 C06ZBQ 118707617 IC50 < 20000 nM T50914 CW2E8V 118707618 IC50 < 20000 nM T50914 CWF9Z6 122189278 IC50 = 215 nM T50914 C5G1MV 122189279 IC50 = 110 nM T94788 CJ3CI2 7168 IC50 > 630957.34 nM T94788 C0X3UH 83254 IC50 = 158489.32 nM T94788 C6TVB7 212827 IC50 = 794328.23 nM T94788 C6DQB5 301729 IC50 > 1258925.41 nM T94788 COWB63 405802 IC50 = 50118.72 nM T94788 CHS6X9 655202 IC50 = 63095.73 nM T94788 C1IZE5 725300 IC50 = 7943.28 nM T94788 CS9J5Y 725306 IC50 = 7943.28 nM T94788 C2CGU9 726159 IC50 = 50118.72 nM T94788 CC6B7T 735015 IC50 = 50118.72 nM T94788 CM56RC 860350 IC50 = 251.19 nM T94788 CDYI60 868259 IC50 = 2511.89 nM T94788 CS2EK8 893481 IC50 = 25118.86 nM T94788 C59MYX 2027971 IC50 = 1258.93 nM T94788 C47BDJ 2776294 IC50 > 1258925.41 nM T94788 C97GYH 3520857 IC50 = 630.96 nM T94788 C2F8XN 3672897 IC50 = 7943.28 nM T94788 CZP8B3 4084523 IC50 > 63095.73 nM T94788 C50KUX 7565541 IC50 = 199526.23 nM T94788 CO4Z6D 8030270 IC50 > 630957.34 nM T94788 C84KXS 9795233 IC50 = 6309.57 nM T94788 C7TFO3 11470832 IC50 = 316227.77 nM T94788 C8O2ZN 12385744 IC50 = 125892.54 nM T94788 CF6VQ0 16770079 IC50 > 1258925.41 nM T94788 C0CUM1 18108101 IC50 > 630957.34 nM T94788 CDWJ60 22374565 IC50 = 158489.32 nM T94788 C5C4BL 26586004 IC50 > 63095.73 nM T94788 CY67FJ 42959251 IC50 > 1258925.41 nM T94788 CH08AN 46360538 IC50 > 63095.73 nM T94788 CVI3P2 68971843 IC50 = 1000000 nM T94788 CD3I4T 78319104 IC50 = 50.12 nM T94788 C6FKA3 91826695 IC50 = 2000 nM T94788 CGD62B 118797287 IC50 = 199.53 nM T94788 CY1C9Z 118797288 IC50 = 1000 nM T94788 CM8L0O 118797289 IC50 = 1995.26 nM T94788 C2UCV5 118988431 IC50 = 50.12 nM T94788 C5D7HA 121231397 IC50 = 1584.89 nM T94788 CV6LN5 122190007 IC50 = 10000 nM T94788 C39SMD 122190008 IC50 = 1258.93 nM T94788 CPE19Z 122190009 IC50 = 251.19 nM T94788 C9FBD1 122190010 IC50 = 199.53 nM T94788 CE07KP 122190011 IC50 = 630.96 nM T94788 CXCS54 122190012 IC50 = 6309.57 nM T94788 CG17JK 122190013 IC50 = 2511.89 nM T94788 C4EV0M 122190014 IC50 = 1995.26 nM T94788 C80GKM 122190015 IC50 = 316.23 nM T94788 CP6K2B 122190016 IC50 = 50.12 nM T94788 C7VS5R 122190017 IC50 = 158.49 nM T94788 C1PTE7 122190018 IC50 = 19.95 nM T94788 C3HK5Z 122190019 IC50 = 1584.89 nM T94788 CI7WO3 122190020 IC50 = 15.85 nM T94788 C4DH0W 122190021 IC50 = 12.59 nM T94788 CTO86S 122190022 IC50 = 50.12 nM T94788 C3YPW8 122190023 IC50 = 31.62 nM T94788 CA81VS 122190024 IC50 = 10 nM T94788 C4F9TM 122190025 IC50 = 794.33 nM T94788 C1Q0LG 122190026 IC50 = 501.19 nM T94788 C57BDC 122190027 IC50 = 501187.23 nM T94788 C50IXQ 122190028 IC50 = 79.43 nM T94788 CX1F3Y 122190029 IC50 = 25.12 nM T94788 C1JN6L 122190030 IC50 = 100 nM T94788 CV6WO5 122190031 IC50 = 1258.93 nM T94788 CSR14P 122190032 IC50 = 199.53 nM T94788 C3VMZ5 122190033 IC50 = 1995.26 nM T94788 CFZ7S6 122190034 IC50 = 630.96 nM T94788 C9RC3A 122190035 IC50 = 3981.07 nM T94788 CW61KB 122190036 IC50 = 31.62 nM T94788 CZ6HV0 122190037 IC50 = 251.19 nM T94788 C74PQW 122190038 IC50 = 1258.93 nM T94788 CJ93MB 122190039 IC50 = 199.53 nM T94788 CFU9D5 122190040 IC50 = 251.19 nM T94788 CE5IU6 122190041 IC50 = 630.96 nM T94788 CN9K6B 122190042 IC50 = 1000 nM T94788 CHYW90 122192294 IC50 > 100000 nM T94788 CWS90E 122192295 IC50 > 100000 nM T94788 C5ZVG8 122192296 IC50 = 74100 nM T94788 C82AYW 122192297 IC50 = 3900 nM T94788 C5FOQ7 122192298 IC50 = 2800 nM T94788 CHY4F9 122192299 IC50 = 15100 nM T94788 C7NWS8 122192300 IC50 = 64600 nM T94788 C0ZAL6 122192301 IC50 > 100000 nM T94788 C6AK1I 122192302 IC50 > 100000 nM T94788 C7L3KO 127028895 IC50 = 3162.28 nM T94788 C4W7VT 127029155 IC50 = 251188.64 nM T94788 C0YEI9 127029156 IC50 > 63095.73 nM T94788 CO3RK0 127029157 IC50 > 63095.73 nM T94788 COG82P 127029167 IC50 = 12589.25 nM T94788 C6C0QA 127029168 IC50 > 63095.73 nM T94788 CP35ME 127030001 IC50 = 1584.89 nM T94788 CV46ES 127031195 IC50 = 15848.93 nM T94788 CSX02I 127031504 IC50 = 10000 nM T94788 CE6YK2 127043627 IC50 = 158.49 nM T94788 CX3KR7 127043628 IC50 = 50.12 nM T94788 C3P2IZ 127043978 IC50 = 630.96 nM T94788 CW5RB9 127043979 IC50 = 501.19 nM T94788 CV6TZ9 127043980 IC50 = 1584.89 nM T94788 CHO9X7 127043981 IC50 = 79.43 nM T94788 CCF9A6 127043987 IC50 = 794.33 nM T94788 CF52GU 127044125 IC50 = 100 nM T94788 CJ4M1D 127044126 IC50 = 630.96 nM T94788 C43FPT 127044127 IC50 = 2511.89 nM T94788 C84POC 127044545 IC50 = 251.19 nM T94788 COX2U0 127044546 IC50 = 251.19 nM T94788 CN2G7O 127044547 IC50 = 1258.93 nM T94788 C8Z0CO 127044548 IC50 = 1995.26 nM T94788 C01DJM 127044549 IC50 = 19952.62 nM T94788 CTI74N 127044550 IC50 = 3162.28 nM T94788 CZW9S7 127044551 IC50 = 2511.89 nM T94788 CT54QC 127044552 IC50 = 1584.89 nM T94788 CXG6Q0 127044553 IC50 = 630.96 nM T94788 C5N2CR 127044723 IC50 = 6309.57 nM T94788 CE9RB2 127044724 IC50 = 1000 nM T94788 C71JPZ 127044725 IC50 = 19952.62 nM T94788 CFRG49 127044726 IC50 = 251.19 nM T98271 D0R0MW 5329102 IC50 = 47.4 nM T98271 CHWL84 6539599 IC50 = 220 nM T98271 C6P4BO 6539600 IC50 = 1200 nM T98271 COD03X 10156251 IC50 = 4.32 nM T98271 C3VRO9 44557921 IC50 = 5888.44 nM T98271 C67OJG 44588117 Ki = 541 nM T98271 CKA12O 57891796 IC50 = 209 nM T98271 C8NF7Y 59699998 IC50 = 23.6 nM T98271 CZ14IK 91938067 IC50 = 0.07 nM T98271 CDL4P0 118009188 IC50 = 3.3 nM T98271 C38SJA 118419786 IC50 = 0.3 nM T98271 CE7L5R 118419870 IC50 = 1400 nM T98271 CS2VP0 118420021 IC50 = 3 nM T98271 CY6NG3 118429629 IC50 = 0.51 nM T98271 CNO6Z1 118429823 IC50 = 0.32 nM T98271 C7YZ8X 118429852 IC50 = 0.42 nM T98271 CJB69T 118429935 IC50 = 0.23 nM T98271 C4H7SM 118714184 IC50 = 319 nM T98271 CR2W8V 118864359 IC50 = 4 nM T98271 CI91CV 121255756 IC50 = 6 nM T98271 CYBU50 124002327 IC50 = 18000 nM T98271 C48IAY 134530903 IC50 = 0.62 nM T98271 C4YWO9 134812845 Ki = 9.1 nM T98271 CG15PY 134812846 Ki = 53000 nM T98271 CQBF40 135284803 IC50 = 0.2 nM T98271 CO58DJ 135390126 IC50 = 886 nM T98271 C6AZ2R 135435018 IC50 = 280 nM T98271 C9O8CQ 137348448 Ki = 8.3 nM T98271 C63TGO 137349551 Ki = 6.3 nM T98271 C6I5ME 137349552 Ki = 10 nM T98271 C1UYP7 137640287 IC50 = 2800 nM T98271 C6B9RI 137655689 IC50 = 350 nM T98271 C0B7LO 138393295 IC50 = 4.02 nM T98271 CYZ4A6 146121078 IC50 = 18000 nM T98271 CRC8D2 155489850 Ki = 78000 nM T98271 CUC56L 155515968 IC50 = 3500 nM T98271 C3W9MD 155516193 IC50 = 9.27 nM T98271 CU9P1O 155516654 IC50 = 72.1 nM T98271 CO79KW 155517221 IC50 = 108 nM T98271 CG8J5X 155518911 Ki = 32 nM T98271 C5OK4J 155519508 IC50 = 3800 nM T98271 CD92PB 155519881 IC50 = 381 nM T98271 C0EH9S 155520094 IC50 = 161 nM T98271 C6Y3ZR 155520697 IC50 = 800 nM T98271 CR3LG7 155520971 IC50 = 420 nM T98271 C4FLT9 155521757 IC50 = 54 nM T98271 CF92OZ 155523797 IC50 = 149 nM T98271 C8YX3N 155525320 IC50 = 910 nM T98271 C1LH3X 155533332 IC50 = 387 nM T98271 CAN08J 155534113 Ki = 20 nM T98271 CHCE71 155534845 IC50 = 3390 nM T98271 C16JRL 155535406 Ki = 33 nM T98271 CX0V3J 155535984 IC50 = 370 nM T98271 C3XR8O 155536206 Ki = 22 nM T98271 CN9MV3 155536780 IC50 = 184 nM T98271 C6VQA5 155537429 IC50 > 50000 nM T98271 CHQN92 155537739 IC50 = 1100 nM T98271 CA74KV 155537883 IC50 = 398 nM T98271 C4G0DY 155538489 IC50 = 4440 nM T98271 CDB8Q3 155540035 IC50 = 381 nM T98271 C8Q4LF 155540633 IC50 = 18.6 nM T98271 CX68YN 155541385 Ki > 100000 nM T98271 CWU67H 155543077 Ki = 30 nM T98271 CBT5A1 155543338 IC50 = 230 nM T98271 CD8K3O 155543384 Ki = 44 nM T98271 C4CV6S 155544989 IC50 = 462 nM T98271 CL51KX 155546156 IC50 = 2200 nM T98271 CUTW39 155546618 Ki = 8.2 nM T98271 C4E0HB 155546757 Ki = 59 nM T98271 CR45OK 155547135 IC50 = 560 nM T98271 C49UVQ 155547733 Ki = 8.5 nM T98271 CI2J4O 155551330 Ki = 22 nM T98271 CM1WS6 155552596 IC50 > 50000 nM T98271 CP2K8O 155554487 Ki = 12 nM T98271 CYC93Q 155556093 IC50 = 612 nM T98271 CS8MC1 155562025 Ki = 39 nM T98271 C8UW4P 155562878 Ki = 6.2 nM T98271 CS7TO0 155566480 IC50 = 120 nM T98271 C53HDP 155568011 IC50 = 71 nM T98271 CMHX39 155568223 IC50 = 7700 nM T98271 CDP94M 155569521 Ki = 24 nM T16739 D07MGA 72281 IC50 = 78760 nM T16739 D0E7PQ 5311 IC50 > 100000 nM T16739 D0H0HJ 19493 IC50 = 4640 nM T16739 D0I9HF 10621 IC50 = 19160 nM T16739 D0K8KX 5280343 IC50 = 1260 nM T16739 D0P9AC 3675 Ki = 5600 nM T16739 D0X9XP 5281613 IC50 = 10140 nM T16739 D04PBH 5280804 IC50 = 950 nM T16739 D05OQG 5318997 IC50 = 26440 nM T16739 D07SDQ 969516 IC50 = 9600 nM T16739 D08EUS 6475492 IC50 = 250 nM T16739 D0I4ZN 66571643 IC50 = 24 nM T16739 D0L0BX 5318980 IC50 = 64490 nM T16739 D0U3EP 445154 IC50 = 10200 nM T16739 D00SUC 74766595 IC50 > 40000 nM T16739 D09NCT 53392492 IC50 = 620000 nM T16739 D08PUW 64982 IC50 = 3550 nM T16739 C2ZB4C 5530 IC50 = 22300 nM T16739 C2N0TD 26070 IC50 = 3600 nM T16739 CD2H6J 147394 IC50 = 4740 nM T16739 CQ3J2T 520838 IC50 > 50000 nM T16739 CIW4B1 654875 IC50 = 25660 nM T16739 C84OLS 681700 IC50 > 188000 nM T16739 CWY8H6 715694 IC50 = 51000 nM T16739 CE04VM 741480 IC50 = 23000 nM T16739 CUP37F 741811 IC50 = 6450 nM T16739 C0RBV2 897193 IC50 > 188000 nM T16739 CIT3L2 1016023 IC50 = 4160 nM T16739 C46ZNQ 1090945 IC50 = 40000 nM T16739 COB92M 1730869 IC50 = 2410 nM T16739 C8SCH5 1797597 IC50 = 18200 nM T16739 CB9RM6 2533167 IC50 > 3000 nM T16739 CY2LD8 2578698 IC50 > 3000 nM T16739 CEQ4V8 2723716 IC50 = 2100 nM T16739 C49LVY 2744807 IC50 = 249000 nM T16739 C05VBZ 2744808 IC50 > 188000 nM T16739 CNP4S1 2806094 IC50 = 1200 nM T16739 C6AF0X 2836494 IC50 = 2800 nM T16739 CTD9P6 2856277 IC50 = 66400 nM T16739 C4DCJ7 3082143 Ki = 188000 nM T16739 CSI96F 3082666 Ki = 79600 nM T16739 CNE29P 3084961 IC50 = 2980 nM T16739 CR7AK6 3132916 IC50 = 51600 nM T16739 CLFE62 3333374 IC50 = 13200 nM T16739 C7E0HC 3701937 IC50 = 3600 nM T16739 CZ0CU8 3945115 IC50 = 19000 nM T16739 CZX1O2 4010130 IC50 = 3600 nM T16739 CMEC57 4539762 IC50 = 26100 nM T16739 CFQ3J7 4779843 IC50 = 34000 nM T16739 CC7R0L 5346910 IC50 = 51400 nM T16739 CIE93U 5777366 IC50 > 3000 nM T16739 CT5NF0 6476700 IC50 = 5000 nM T16739 C5YT8F 6611223 IC50 = 7580 nM T16739 C1MD3E 6614843 IC50 = 870 nM T16739 CW25IO 6759146 IC50 = 300 nM T16739 C23BXN 6759311 IC50 = 3100 nM T16739 CT0PW1 6787939 IC50 = 550 nM T16739 CL0OZ9 9606714 IC50 > 3000 nM T16739 COBY28 9664194 IC50 > 10000 nM T16739 C3I9EM 9918200 IC50 = 500 nM T16739 CP0X9Z 10442008 Ki = 41800 nM T16739 CAC7U5 10666499 IC50 = 50500 nM T16739 CI2QH8 10910111 IC50 > 100000 nM T16739 CIR64S 11016019 IC50 = 21830 nM T16739 CG16JP 11543975 IC50 > 10000 nM T16739 C9K2ZQ 12106307 IC50 > 100000 nM T16739 CP48AH 12450112 IC50 = 77500 nM T16739 C2PEQ9 12915214 IC50 = 882.3 nM T16739 C4EH5W 12915218 IC50 > 10000 nM T16739 C8ANC5 13380562 IC50 = 15600 nM T16739 CO67NT 13559597 IC50 = 5600 nM T16739 CK08BO 13896866 IC50 = 30000 nM T16739 CEJZ38 16047167 IC50 = 500 nM T16739 CB78XP 16047280 IC50 = 1000 nM T16739 CZU6D2 16368147 IC50 = 20300 nM T16739 CJ0I9K 19203678 IC50 = 49200 nM T16739 CEUV82 24632452 IC50 > 188000 nM T16739 CDVA38 25045938 IC50 = 16600 nM T16739 CF47JU 25138011 IC50 > 100000 nM T16739 C92TFZ 25335287 IC50 = 13700 nM T16739 CSC9F8 25501843 IC50 = 37700 nM T16739 C0GAW5 36217788 Ki = 3700 nM T16739 CMEI72 39243036 Ki = 8900 nM T16739 C7C6BT 39243042 IC50 = 3700 nM T16739 C8MCW0 43343228 IC50 = 111400 nM T16739 C5SR1T 43810345 Ki = 8000 nM T16739 CJ8ZA4 44572695 IC50 = 321.1 nM T16739 CV21MX 44577626 IC50 = 2100 nM T16739 CL2TP4 44577718 IC50 > 25000 nM T16739 CU6S7O 44607264 IC50 = 2500 nM T16739 C1CT7A 44607267 IC50 = 9700 nM T16739 CS29ZA 45376216 IC50 = 25 nM T16739 C1JEG9 46236753 IC50 = 21 nM T16739 CS3L6B 46236755 Ki = 1300 nM T16739 C6JUK7 46830228 IC50 = 150 nM T16739 C1FN3T 46830229 Ki = 1000 nM T16739 CR0I8A 46830231 Ki = 1000 nM T16739 C72IST 46830246 IC50 = 19 nM T16739 CZ3F2M 46830247 Ki = 1000 nM T16739 C4FAU9 46868342 IC50 = 19500 nM T16739 CY9MF4 46868344 IC50 = 14000 nM T16739 CS6W7J 46889939 IC50 = 13000 nM T16739 C82MIK 46988215 IC50 = 58800 nM T16739 C52UHN 49864177 IC50 = 1900 nM T16739 C35XSM 49868483 Ki = 610 nM T16739 C8DEO9 53258076 IC50 = 1600 nM T16739 CY0IU1 53258078 IC50 = 6700 nM T16739 CDX7H2 53842276 Ki > 100000 nM T16739 CAG3F4 55285162 IC50 = 1720 nM T16739 CKA1L9 56653684 IC50 = 20 nM T16739 C32VWF 56659548 IC50 = 9000 nM T16739 C0JWZ4 56660074 Ki = 6800 nM T16739 CIU3D9 56662993 Ki = 8900 nM T16739 CD57TH 56666474 Ki = 1800 nM T16739 C8VI0Z 56670425 Ki = 11700 nM T16739 CF92TL 56670426 Ki = 2000 nM T16739 CK8I6H 56673395 IC50 = 9000 nM T16739 CFYW34 56673396 Ki = 1500 nM T16739 CVX90D 56673911 Ki = 6000 nM T16739 C62MVT 56683888 Ki > 100000 nM T16739 C73OFQ 56943211 IC50 = 16800 nM T16739 CG5N1V 57397741 Ki = 9 nM T16739 CJ3RM8 57402930 Ki = 5 nM T16739 C3NUX4 60149007 IC50 = 8 nM T16739 C68XHY 60161811 IC50 = 70 nM T16739 CA2LX1 60166618 IC50 > 10000 nM T16739 CD6B5P 60203904 IC50 = 62 nM T16739 CL0M4Y 62999067 IC50 > 188000 nM T16739 C4AR3Y 64545027 IC50 > 188000 nM T16739 CQTC83 66571530 IC50 = 5 nM T16739 CCO53I 66571532 IC50 = 6 nM T16739 CS7ZX1 66571590 IC50 = 6 nM T16739 CB6CU0 66630014 IC50 = 20 nM T16739 C18MPL 70723639 IC50 = 210 nM T16739 CC6QA0 71458817 Ki = 610 nM T16739 CJP68B 71543365 EC50 = 0.95 nM T16739 C8XZ7O 71554173 IC50 = 18 nM T16739 CSM4W0 71616357 IC50 = 8000 nM T16739 CH0I3Z 71616358 IC50 = 56500 nM T16739 C2PKM3 71616359 IC50 = 69200 nM T16739 CQ3I9J 71616361 IC50 = 2100 nM T16739 CJF4I0 71616469 IC50 = 18400 nM T16739 C3YL4O 71616470 IC50 > 125000 nM T16739 C8F9HJ 71616471 IC50 = 88900 nM T16739 C8F4IT 71616472 IC50 = 19000 nM T16739 CL4PU5 71616473 IC50 = 51200 nM T16739 CPNY67 71616589 IC50 > 125000 nM T16739 CQ05ZS 71616591 IC50 > 125000 nM T16739 C7IP1M 71616593 IC50 > 125000 nM T16739 C5HPG0 71652824 IC50 = 390 nM T16739 CDN0A9 71652976 IC50 = 21600 nM T16739 C10VWG 71652977 IC50 = 11500 nM T16739 CW9E3M 71652978 IC50 = 17300 nM T16739 C57LZP 71652979 IC50 = 69300 nM T16739 CH8Z3K 71652980 IC50 > 125000 nM T16739 C0MI9R 71652981 IC50 > 125000 nM T16739 CNI6L9 71652982 IC50 = 28900 nM T16739 C3QNB6 71653121 IC50 = 19500 nM T16739 CEO2Y0 71653122 IC50 > 125000 nM T16739 CRP27T 71653123 IC50 > 125000 nM T16739 CE3N2H 71653124 IC50 = 32800 nM T16739 CF40MB 71653125 IC50 = 47600 nM T16739 C6FB9D 71653126 IC50 = 53200 nM T16739 CWBS20 71653266 IC50 > 125000 nM T16739 C1TG6A 71653267 IC50 = 22400 nM T16739 C37CMZ 71653268 IC50 = 35100 nM T16739 C14QWL 71653269 IC50 = 29500 nM T16739 CB81FJ 71653270 IC50 = 43500 nM T16739 CJ7UZ9 71653425 IC50 > 125000 nM T16739 C6M9RH 71653426 IC50 > 125000 nM T16739 C4GMJ9 71653427 IC50 > 125000 nM T16739 CCS5N8 71663254 IC50 = 9500 nM T16739 C07XGC 71664305 IC50 = 11.26 nM T16739 C6PV0U 71760961 IC50 > 125000 nM T16739 CKU7B3 72713113 IC50 > 125000 nM T16739 CE41SJ 72713114 IC50 > 125000 nM T16739 CMC6L0 72713115 IC50 = 43300 nM T16739 C7DM0N 72713116 IC50 > 125000 nM T16739 C9FRJ3 72713117 IC50 > 125000 nM T16739 C0UX4C 72713118 IC50 = 27500 nM T16739 C3DPJ6 72713319 IC50 = 70700 nM T16739 CY72VF 72713320 IC50 > 125000 nM T16739 C7BZ5U 72713321 IC50 = 77100 nM T16739 CK8P3Z 72713322 IC50 = 81300 nM T16739 C26IKX 72713323 IC50 > 125000 nM T16739 C72YQH 72713324 IC50 > 125000 nM T16739 C5PVG2 72713325 IC50 = 87400 nM T16739 CS0C1O 72713326 IC50 = 17000 nM T16739 CO65IU 72713327 IC50 = 15000 nM T16739 CR19YB 72713328 IC50 = 30200 nM T16739 CGL54S 72713329 IC50 = 47100 nM T16739 CF1UM3 72713330 IC50 = 25300 nM T16739 C7C8VE 72713537 IC50 > 125000 nM T16739 CE9HF5 72713538 IC50 > 125000 nM T16739 C53VFH 72713539 IC50 > 125000 nM T16739 C8XI3V 72713540 IC50 > 125000 nM T16739 C4J8QH 72713541 IC50 > 125000 nM T16739 C1T4XR 72713542 IC50 > 125000 nM T16739 COIN32 72713758 IC50 > 125000 nM T16739 CB83MO 72713759 IC50 > 125000 nM T16739 CCR68V 72713760 IC50 > 125000 nM T16739 C54CMZ 72713761 IC50 > 125000 nM T16739 CRI35G 72713762 IC50 > 125000 nM T16739 CMA2E7 72713763 IC50 > 125000 nM T16739 C0Q9UJ 72713972 IC50 = 83400 nM T16739 CGL9V5 72713973 IC50 = 100100 nM T16739 C7CTX5 72713974 IC50 > 125000 nM T16739 CG01AT 72713975 IC50 = 40300 nM T16739 CL98ZG 72713976 IC50 > 125000 nM T16739 CI7WS4 72713977 IC50 > 125000 nM T16739 C6MA9B 72714188 IC50 > 125000 nM T16739 CWC3T5 72714189 IC50 > 125000 nM T16739 CLVI57 72714190 IC50 > 125000 nM T16739 CEK73N 72714191 IC50 > 125000 nM T16739 CY72LF 72714192 IC50 > 125000 nM T16739 CBE35Y 72714193 IC50 > 125000 nM T16739 CEX81W 72714194 IC50 > 125000 nM T16739 C7JA5Z 72714195 IC50 > 125000 nM T16739 C5JP7I 72714196 IC50 = 27600 nM T16739 C2YD3U 72714197 IC50 = 39800 nM T16739 CS3AP6 72714198 IC50 = 43900 nM T16739 CN3KI1 72714199 IC50 = 35700 nM T16739 CF0YT9 72714200 IC50 = 45700 nM T16739 CGK06E 72714201 IC50 = 55100 nM T16739 C3TGI7 72792551 IC50 > 3000 nM T16739 C9E3XN 72792612 IC50 > 3000 nM T16739 CHDB60 72793898 EC50 = 62 nM T16739 CK7Q5I 72856745 IC50 = 17200 nM T16739 CEIQ48 73055052 IC50 = 670 nM T16739 CGY9Z7 73055053 IC50 = 84200 nM T16739 C4L8AF 73055054 IC50 = 10330 nM T16739 C6DR0Q 73055333 IC50 = 810 nM T16739 C6I0VD 73055334 IC50 = 530 nM T16739 C5XR9V 73055335 IC50 = 710 nM T16739 C9QGE8 73055336 IC50 = 3000 nM T16739 CY14US 73055337 IC50 = 830 nM T16739 C27MKG 73055636 IC50 = 102560 nM T16739 CRP05T 73334474 IC50 = 143600 nM T16739 CUN26K 73334475 IC50 = 131900 nM T16739 CS36LK 73334584 IC50 = 184200 nM T16739 C81IEB 73334585 IC50 = 93100 nM T16739 CS79XE 73334588 IC50 = 51700 nM T16739 CZ58FD 73334589 IC50 = 92200 nM T16739 CV5JY9 73334590 IC50 = 22200 nM T16739 CPG73S 73417116 IC50 < 2000 nM T16739 CI9Q0G 76281715 IC50 = 300 nM T16739 C05TJO 76282229 IC50 = 480 nM T16739 CC5IG0 76282703 IC50 = 580 nM T16739 CA8YE3 76282705 IC50 = 410 nM T16739 C68RKH 76310231 IC50 < 1000 nM T16739 CVJW69 76311323 IC50 = 76050 nM T16739 CF4YT3 76311324 IC50 = 18100 nM T16739 C70MNC 76311325 IC50 = 17300 nM T16739 C3N4EY 76311326 IC50 = 19300 nM T16739 CP8L3T 76311327 IC50 = 29500 nM T16739 CCS6N0 76313844 IC50 > 3000 nM T16739 C94ARC 76313846 IC50 = 1900 nM T16739 C51KFJ 76313916 Ki = 9 nM T16739 C20FBC 76314915 IC50 > 188000 nM T16739 CK53JN 76314916 IC50 = 7500 nM T16739 C83COP 76314917 IC50 = 27800 nM T16739 C4TCX5 76314918 IC50 = 34900 nM T16739 CO1EN3 76317452 IC50 = 2200 nM T16739 CJ5KN9 76318471 IC50 > 125000 nM T16739 CD1K3Y 76318528 IC50 > 188000 nM T16739 C4KLE9 76318530 IC50 = 44400 nM T16739 C9KG2U 76318531 IC50 > 188000 nM T16739 CC50ZL 76318532 IC50 = 26300 nM T16739 CV9MQ4 76318533 IC50 = 16200 nM T16739 CT5FZ8 76321184 IC50 < 1000 nM T16739 C6XRT0 76321186 IC50 < 1000 nM T16739 CX91NY 76322188 IC50 = 57000 nM T16739 CT8JY2 76322189 IC50 = 36100 nM T16739 CWCI08 76322190 IC50 = 10200 nM T16739 CTH0U1 76322191 IC50 = 19000 nM T16739 C83GJS 76322192 IC50 = 29600 nM T16739 C0C1ZL 76324746 IC50 = 12000 nM T16739 C7K3MB 76324808 Ki = 5 nM T16739 CA0X3B 76325809 IC50 = 13700 nM T16739 CU9I8M 76325810 IC50 = 13700 nM T16739 CKB5O9 76328366 IC50 = 1000 nM T16739 CZQ1P0 76329344 IC50 > 125000 nM T16739 CPJ39A 76329395 IC50 > 188000 nM T16739 CD0OG4 76329396 IC50 = 43200 nM T16739 CCU16Y 76329397 IC50 = 17200 nM T16739 C0NL9S 76329398 IC50 = 43600 nM T16739 CN34ZA 76329399 IC50 = 40100 nM T16739 CWK86G 76329400 IC50 = 61600 nM T16739 CUY96G 76329401 IC50 = 23600 nM T16739 C3PHJ5 76329402 IC50 = 26000 nM T16739 CBL71T 76333040 IC50 = 123000 nM T16739 CM5OJ0 76333041 IC50 = 26900 nM T16739 CO14DA 76333043 IC50 = 85700 nM T16739 CHRQ49 76333044 IC50 > 188000 nM T16739 C10HPW 76333045 IC50 = 15800 nM T16739 CXG5C1 76333046 IC50 = 10300 nM T16739 C4I0PD 76333047 IC50 = 9500 nM T16739 CV1P3Z 76333048 IC50 = 17500 nM T16739 CK0SM6 76333049 IC50 = 56900 nM T16739 CPT6Q2 76335554 IC50 = 5200 nM T16739 CUNK03 76335652 IC50 = 1600 nM T16739 CFAW05 76336591 IC50 > 125000 nM T16739 CE6W9D 76336592 IC50 > 125000 nM T16739 CR16LQ 76336665 IC50 > 188000 nM T16739 C3TW1I 76336666 IC50 = 17600 nM T16739 C34RKL 76336667 IC50 = 12900 nM T16739 CG5Z1U 77014306 Ki = 59 nM T16739 C02JLH 86273745 IC50 < 1000 nM T16739 CC7U0M 86278919 IC50 = 610 nM T16739 C4KZU2 86343599 IC50 = 21250 nM T16739 C74WUO 86729878 IC50 = 30 nM T16739 CJ64QM 86729882 IC50 = 50 nM T16739 C4O6WM 87056304 IC50 = 41495.4 nM T16739 C2AJ5M 87056305 IC50 = 4880 nM T16739 C2WOA8 87056306 IC50 = 3160 nM T16739 C9AO8E 87056307 IC50 = 11190 nM T16739 C4GO8Z 87056308 IC50 = 5060 nM T16739 COI6M2 87056309 IC50 > 125000 nM T16739 CH8EW4 87057268 IC50 = 45708.82 nM T16739 CV85ZS 87057352 IC50 = 8330 nM T16739 C16LNO 87057353 IC50 = 3130 nM T16739 CD09YU 87057354 IC50 = 24370 nM T16739 CP3EQ4 87057355 IC50 = 24710 nM T16739 CJRB81 87057356 IC50 = 26480 nM T16739 CMJ09Y 87057357 IC50 = 21820 nM T16739 CZM8B9 87057358 IC50 = 59160 nM T16739 CXLW25 87057359 IC50 = 125025.9 nM T16739 C78HFR 87057441 IC50 > 125000 nM T16739 C4UR3X 87057443 IC50 = 1590 nM T16739 C4I9QR 87057444 IC50 = 1590 nM T16739 C4YE0G 87057445 IC50 = 650 nM T16739 CQV6O1 87057446 IC50 = 1660 nM T16739 C91RJF 87057447 IC50 = 1590 nM T16739 CDHM84 87057448 IC50 = 1080 nM T16739 C6JM8W 87057533 IC50 = 1100 nM T16739 CY83SD 87057534 IC50 = 2580 nM T16739 C3HEA2 87057535 IC50 = 3580 nM T16739 CS2U9C 87057537 IC50 = 2610 nM T16739 CKAD16 87057538 IC50 = 7400 nM T16739 CHZ78V 87057539 IC50 = 2640 nM T16739 CQV8P5 90197341 IC50 = 9132 nM T16739 CAE9S6 90197458 IC50 = 975 nM T16739 C97DGB 90197459 IC50 = 779 nM T16739 CP4FQ2 90197685 IC50 = 584 nM T16739 CB2RV3 90197737 IC50 = 335 nM T16739 CJW98L 90197739 IC50 = 617 nM T16739 C6AK9N 90197969 IC50 = 608 nM T16739 C2J9PM 90665012 IC50 = 100 nM T16739 C1KQ7P 91971954 IC50 = 230 nM T16739 CU5D3W 93990915 IC50 = 66.1 nM T16739 C7RTD0 101927272 IC50 = 22000 nM T16739 CS1Q4M 102101183 IC50 = 800 nM T16739 CV3E5J 102101190 IC50 = 8400 nM T16739 CI1Q0T 102197009 IC50 = 10100 nM T16739 CWX5P2 102300629 IC50 = 100.2 nM T16739 CFT89B 102313433 IC50 = 2400 nM T16739 C3RW4H 102313434 IC50 = 380 nM T16739 C2S1AO 110264830 IC50 > 25000 nM T16739 CMQ4A7 117926025 IC50 = 90000 nM T16739 CIDX08 118152103 IC50 < 10 nM T16739 CBT5S7 118290227 IC50 < 100 nM T16739 C4UK8C 118290492 IC50 < 100 nM T16739 CATK81 118292440 IC50 < 100 nM T16739 C61BNV 118304877 IC50 < 1000 nM T16739 CKD37J 118432652 IC50 < 100 nM T16739 C1VB4J 118432667 IC50 < 100 nM T16739 C1MUS4 118432683 IC50 = 180 nM T16739 C2M5CU 118432730 IC50 < 100 nM T16739 C2YPX9 118432772 IC50 = 210 nM T16739 CM56VT 118432893 IC50 = 240 nM T16739 CYM0B5 118433105 IC50 < 100 nM T16739 C2U3NT 118483746 IC50 = 3260 nM T16739 C38WNG 118483913 IC50 = 131 nM T16739 C6A8FW 118483914 IC50 = 161 nM T16739 CF7Z1S 118493308 IC50 < 100 nM T16739 C6Q3JH 118626619 EC50 = 59 nM T16739 C4OAM2 118626625 EC50 = 110 nM T16739 CD6IW9 118626626 IC50 = 3 nM T16739 CSA0H4 118626627 EC50 = 27 nM T16739 CWA4U7 118626659 EC50 = 160 nM T16739 CO2U6F 118626664 EC50 = 59 nM T16739 CQ3H6M 118626669 IC50 = 18 nM T16739 C71RFN 118626673 EC50 = 47 nM T16739 C3SX8V 118626689 EC50 = 100 nM T16739 CT3M1R 118626694 EC50 = 22 nM T16739 CZNA53 118626736 EC50 = 14 nM T16739 C4V1YJ 118626744 EC50 = 13 nM T16739 CAW87G 118626755 EC50 = 45 nM T16739 C72BEP 118626766 EC50 = 150 nM T16739 CI4RV0 118626770 IC50 = 4 nM T16739 CWU97Y 118626775 EC50 = 34 nM T16739 CZC1R5 118626784 EC50 = 66 nM T16739 CQNL01 118642942 EC50 = 43 nM T16739 C4H1TQ 118712953 IC50 = 358 nM T16739 C4J8TS 118712954 IC50 = 218 nM T16739 CH0YP2 118712955 IC50 = 202 nM T16739 C2BZ4I 118712956 IC50 = 1780 nM T16739 C64XRP 118713036 IC50 > 125000 nM T16739 CW3X1O 118713037 IC50 > 125000 nM T16739 CZ2SE8 118713038 IC50 > 125000 nM T16739 C5CDL0 118713039 IC50 = 125000 nM T16739 CQ9G6P 118713040 IC50 > 125000 nM T16739 CH7Y8I 118718071 IC50 = 990 nM T16739 CU6CA2 118718080 IC50 = 5000 nM T16739 CFWJ56 118728390 IC50 = 8000 nM T16739 CMEA81 118728391 IC50 = 7000 nM T16739 CJ8ZY2 118728392 Ki = 2400 nM T16739 CW8Z2H 118728853 IC50 = 148 nM T16739 C9XEY8 118728854 IC50 = 223 nM T16739 CVCT10 118728855 IC50 = 11000 nM T16739 C1JX3S 118728856 IC50 = 283 nM T16739 CULF09 118728857 IC50 > 100000 nM T16739 CDKA92 118728858 IC50 = 88000 nM T16739 C4XUG3 118728859 IC50 = 158 nM T16739 CK3E9J 118728860 IC50 = 356 nM T16739 C8L6TZ 118728861 IC50 = 443 nM T16739 CS8UI6 118728862 IC50 > 10000 nM T16739 C90IAX 118733202 IC50 = 1080 nM T16739 C6UT4F 118733203 IC50 = 1820 nM T16739 C6DFB3 118733204 IC50 = 4880 nM T16739 CU0PW1 118733310 IC50 = 125000 nM T16739 CU7H0W 118733311 IC50 = 124671 nM T16739 CMG8V1 118733312 IC50 > 125000 nM T16739 CTW9L7 118733313 IC50 > 125000 nM T16739 C8N2VP 118733314 IC50 > 125000 nM T16739 C8PUK6 118733315 IC50 > 125000 nM T16739 C1LKP9 118733316 IC50 > 125000 nM T16739 CR1Y9S 118733317 IC50 > 125000 nM T16739 C5I0GQ 118733318 IC50 = 26480 nM T16739 C6THG7 118733319 IC50 = 97296 nM T16739 CZ8M9A 118733320 IC50 = 125000 nM T16739 C2JLD1 118733321 IC50 = 98174.79 nM T16739 C48GJF 118733322 IC50 = 125000 nM T16739 C6RY3J 118734094 IC50 = 13 nM T16739 CY57TV 118734096 IC50 = 11690 nM T16739 C0SR8X 118734098 IC50 = 10890 nM T16739 CIW4G9 118734100 IC50 = 74650 nM T16739 C0J2WE 118734102 IC50 = 26 nM T16739 CW81OF 118734104 IC50 = 22 nM T16739 CCN86A 118734106 IC50 = 2730 nM T16739 CH7OT9 118734108 IC50 = 450 nM T16739 C7Y0LX 118735096 IC50 = 360 nM T16739 C8QOE4 118735098 IC50 = 390 nM T16739 CJVK69 119081409 IC50 > 25000 nM T16739 CW5K4Q 122629343 IC50 < 100 nM T16739 CM41DK 126824881 IC50 = 4070 nM T16739 C07AWO 127024901 Ki > 50000 nM T16739 CDGK48 127024902 Ki > 50000 nM T16739 C2WJ8O 127024903 Ki = 22300 nM T16739 CLE3A4 127024904 Ki > 50000 nM T16739 CA2N3H 127024905 Ki = 43800 nM T16739 CD96WJ 127024906 Ki = 7600 nM T16739 C5JR8X 127024910 Ki = 220 nM T16739 C6L9NO 127024911 Ki = 150 nM T16739 C5VA3K 127024912 Ki = 4900 nM T16739 CEP6I1 127024913 Ki = 1200 nM T16739 CX8CQ1 127024953 Ki = 540 nM T16739 CS41MI 127024954 Ki = 16500 nM T16739 C1HC8M 127024955 Ki > 50000 nM T16739 C1GNS7 127025220 Ki > 50000 nM T16739 CBFR58 127025221 Ki > 50000 nM T16739 C15ABD 127025225 IC50 = 77 nM T16739 CO8H3N 127025530 Ki > 50000 nM T16739 C71TYR 127025531 Ki = 47800 nM T16739 CMX37U 127026390 Ki > 50000 nM T16739 C21FPK 127026447 Ki = 32200 nM T16739 CA5P3C 127026448 Ki = 26200 nM T16739 C1HE5A 127026449 Ki = 9100 nM T16739 C6LO3W 127026686 Ki = 650 nM T16739 C81XFS 127027035 Ki = 4000 nM T16739 CO03AZ 127027036 Ki = 220 nM T16739 CU04XV 127027037 Ki = 570 nM T16739 CF2PB5 127027038 Ki = 1200 nM T16739 CNR05U 127027039 Ki = 58 nM T16739 C8WJF6 127027348 Ki = 29 nM T16739 CM57WD 127027349 Ki = 800 nM T16739 C51ULJ 127027685 Ki = 200 nM T16739 CPGJ91 127028003 Ki = 88 nM T16739 C1ZXG0 127028004 Ki = 740 nM T16739 C5A9ZJ 127028005 Ki = 46 nM T16739 C7EO1G 127028006 Ki = 5000 nM T16739 C69TFU 127028007 Ki = 3200 nM T16739 C9HR1P 127028008 Ki = 1800 nM T16739 C5IGO0 127028297 Ki = 1800 nM T16739 C9EK5U 127028662 Ki = 380 nM T16739 CS4G3Z 127028663 Ki = 2400 nM T16739 C9U6ZG 127028664 Ki > 50000 nM T16739 CHB3T4 127028981 Ki > 50000 nM T16739 CY2J0O 127028982 Ki > 50000 nM T16739 C7LP2I 127028983 Ki > 50000 nM T16739 C9DY4H 127030057 Ki = 1800 nM T16739 CS93HT 127030355 Ki = 210 nM T16739 C9O7MN 127030710 Ki = 8000 nM T16739 CF01PG 127030948 Ki = 240 nM T16739 C3FJ9D 127030986 IC50 < 100 nM T16739 CDL0C7 127031303 IC50 = 132 nM T16739 C1LBS7 127031599 Ki = 28400 nM T16739 CGJ45P 127031600 Ki = 2600 nM T16739 CR7LQ2 127032104 Ki = 140 nM T16739 CKYD38 127052923 IC50 = 3180 nM T16739 CA1L0G 129216206 IC50 = 90 nM T16739 CLB30F 130201615 IC50 = 3 nM T16739 CQ0L5P 130901691 IC50 > 25000 nM T16739 CP8L7V 132137973 IC50 = 4090 nM T16739 CRG1Y4 132342060 IC50 = 5600 nM T16739 CZH0Y7 132547265 Ki = 1600 nM T16739 CWQJ96 132547266 Ki > 300000 nM T16739 CYX37Z 134131047 Ki = 190000 nM T16739 CZ34KT 134395060 IC50 = 4 nM T16739 CB13SU 134395087 IC50 = 3 nM T16739 CYC35I 134395111 IC50 = 4 nM T16739 CR2V8E 135326422 EC50 = 68 nM T16739 C9KL2E 135326441 EC50 = 110 nM T16739 CDX54R 135326463 IC50 = 16 nM T16739 CV37UB 135326482 IC50 = 10 nM T16739 CN1LH8 135326483 EC50 = 8 nM T16739 CW8BG2 135400291 IC50 = 275 nM T16739 C3G1IP 135412162 IC50 = 196 nM T16739 C1E9ZN 135442596 IC50 = 291 nM T16739 C5XR3V 135478291 IC50 = 6420 nM T16739 C1N6QZ 135478386 IC50 = 333 nM T16739 C9UZX8 135578375 IC50 = 128 nM T16739 CCNH91 135743577 Ki = 13.5 nM T16739 CZ97SK 135778696 IC50 = 218 nM T16739 CS29LX 135859840 IC50 > 100000 nM T16739 C8B4RF 135905415 IC50 = 98 nM T16739 CX9W4T 136179193 IC50 = 1100 nM T16739 C7O2NJ 136224203 IC50 > 3000 nM T16739 CM06DY 136240105 IC50 = 19 nM T16739 CAB79P 136241665 IC50 = 40 nM T16739 C6DS9L 136245080 IC50 > 3000 nM T16739 CA3P9K 136249363 IC50 > 3000 nM T16739 C5MD2W 136264445 IC50 = 14 nM T16739 CI1PG4 136264446 IC50 > 3000 nM T16739 C96DBR 136264447 IC50 > 3000 nM T16739 CGX86F 137060470 IC50 = 9.2 nM T16739 CS0J7C 137060471 IC50 = 1.7 nM T16739 CO04UM 137375909 IC50 = 9 nM T16739 CGJ2A1 137631451 IC50 = 290 nM T16739 CF5ZR4 137631816 IC50 = 758 nM T16739 CV2O6D 137631867 IC50 = 717 nM T16739 C4R8VL 137632175 IC50 = 720 nM T16739 CUO8Q7 137632382 IC50 = 739.11 nM T16739 CXL78Z 137632856 IC50 > 50000 nM T16739 CP8JC3 137633372 IC50 > 30000 nM T16739 C15LZP 137633523 IC50 = 6300 nM T16739 CVI73M 137633548 IC50 > 10000 nM T16739 C4LU6O 137633775 IC50 = 480 nM T16739 C3J9AI 137633935 IC50 = 210 nM T16739 CDU72C 137633963 IC50 = 340 nM T16739 C42DZX 137634067 IC50 > 10000 nM T16739 CAW57J 137634265 IC50 = 678 nM T16739 CB31GP 137634468 IC50 > 30000 nM T16739 C7X1KG 137634820 IC50 = 3610 nM T16739 CT6GZ3 137634907 IC50 > 10000 nM T16739 CJ03QE 137634970 IC50 > 10000 nM T16739 C41LEK 137635428 IC50 = 210.02 nM T16739 C4QDO2 137635634 IC50 > 10000 nM T16739 C8JDR3 137635678 IC50 > 10000 nM T16739 C2RVD6 137635741 IC50 = 5700 nM T16739 CDE25V 137635795 IC50 = 430 nM T16739 C67IZH 137635859 IC50 > 25000 nM T16739 CP31TR 137636128 IC50 > 10000 nM T16739 CNYO52 137636664 IC50 = 510 nM T16739 CRC52W 137636687 IC50 = 4400 nM T16739 C3P6FE 137637077 IC50 = 2800 nM T16739 CQ26LK 137637420 IC50 = 7600 nM T16739 CPO69Y 137637991 Ki = 30 nM T16739 CUL8I3 137637996 IC50 > 25000 nM T16739 CED9X0 137638271 IC50 = 1300 nM T16739 CVY2J4 137638282 IC50 = 11900 nM T16739 C07ECJ 137638988 IC50 > 50000 nM T16739 CZS28N 137639034 IC50 > 150000 nM T16739 CY6VP5 137639127 IC50 = 57 nM T16739 CVMS92 137639487 IC50 = 123.86 nM T16739 CDLX68 137639830 Ki > 500000 nM T16739 CF38JX 137639972 IC50 > 50000 nM T16739 C46OFJ 137640007 IC50 = 333.54 nM T16739 C68TJS 137640148 IC50 > 10000 nM T16739 CKVY47 137640483 IC50 = 830 nM T16739 CVU6G8 137640490 IC50 = 1600 nM T16739 CQ3P6J 137640719 IC50 > 10000 nM T16739 C6IL1K 137640761 IC50 = 960 nM T16739 CA7K3N 137640895 IC50 = 12600 nM T16739 CI0X1S 137640925 IC50 = 83 nM T16739 CAV75P 137641024 IC50 > 50000 nM T16739 C3WI0J 137641032 IC50 = 170 nM T16739 CQL08Y 137641137 IC50 = 1500 nM T16739 CLS5W8 137641585 IC50 > 10000 nM T16739 C14UKH 137641639 IC50 = 192.93 nM T16739 C6PSJ5 137641751 IC50 = 15600 nM T16739 CRP2C0 137642053 IC50 = 570 nM T16739 C0PM9C 137642315 IC50 = 557 nM T16739 CPL17B 137642483 IC50 > 30000 nM T16739 C2Q3GI 137643093 Ki = 40 nM T16739 C1Y9GT 137643447 IC50 = 1200 nM T16739 C37NTM 137643555 Ki = 290 nM T16739 CK64CO 137643664 IC50 = 270 nM T16739 CGU69C 137643923 IC50 = 200 nM T16739 C5GSD8 137644007 IC50 > 10000 nM T16739 CUN34T 137644037 IC50 = 564 nM T16739 CX3E4R 137644112 IC50 > 25000 nM T16739 CY8HA2 137644280 IC50 = 2600 nM T16739 CJM6D3 137644455 Ki = 380 nM T16739 CMVY45 137644507 IC50 > 50000 nM T16739 CQ0CK5 137644883 IC50 > 50000 nM T16739 CT1QL6 137645063 IC50 = 685 nM T16739 CHP7O4 137645096 IC50 = 1300 nM T16739 CSLK78 137645133 IC50 > 50000 nM T16739 C3AVZ0 137645374 IC50 = 4100 nM T16739 CVCE72 137645494 Ki = 170000 nM T16739 C0ERJ6 137645766 IC50 > 10000 nM T16739 C13GPJ 137645789 IC50 > 10000 nM T16739 C48DHO 137646074 IC50 = 5200 nM T16739 CQ9Y7O 137646081 IC50 = 16000 nM T16739 CL97VA 137646171 IC50 = 6700 nM T16739 C0IHG3 137646527 IC50 > 10000 nM T16739 C2YA8I 137646650 IC50 = 2590 nM T16739 C0NWV1 137647092 EC50 = 300 nM T16739 CD9R0S 137647138 IC50 > 10000 nM T16739 C9YDG1 137647202 IC50 = 680 nM T16739 C38CZQ 137647309 IC50 = 990 nM T16739 CU4JN5 137647385 Ki > 500000 nM T16739 C54NIV 137647590 Ki = 1400 nM T16739 COBV90 137647701 IC50 = 710 nM T16739 C3X8JA 137647705 IC50 > 25000 nM T16739 C8XJ7A 137647789 IC50 = 9000 nM T16739 CJY59L 137647936 Ki = 6300 nM T16739 CX12ZW 137648278 IC50 = 1200 nM T16739 CAU5M1 137648395 IC50 = 13100 nM T16739 CY1HO0 137648656 IC50 > 10000 nM T16739 CX48EV 137648716 IC50 = 750 nM T16739 C8GO0J 137648751 IC50 = 391.15 nM T16739 CMBT98 137648914 IC50 = 16400 nM T16739 CTO60S 137648992 IC50 = 2600 nM T16739 C7Z8CU 137650441 IC50 = 150 nM T16739 CD1JZ6 137650599 IC50 = 1200 nM T16739 C1AC7Q 137650930 IC50 > 50000 nM T16739 CYTE60 137651513 IC50 = 4100 nM T16739 CD8HB9 137651608 IC50 = 9200 nM T16739 CUXY13 137651912 IC50 = 410 nM T16739 CO02PT 137651988 IC50 = 8200 nM T16739 C0U6LH 137652118 IC50 = 30000 nM T16739 C3G4DT 137652360 IC50 = 670 nM T16739 CQ61OF 137652397 IC50 = 24300 nM T16739 CC1TL4 137652408 IC50 = 3000 nM T16739 CKW9B5 137652423 IC50 = 810 nM T16739 C6AY7B 137652448 IC50 > 10000 nM T16739 CA3QK7 137652917 IC50 = 2600 nM T16739 C63JEA 137653002 IC50 = 260 nM T16739 CHO54U 137653055 IC50 = 5200 nM T16739 C81MPW 137653612 IC50 = 650 nM T16739 C80RBG 137653644 Ki = 9800 nM T16739 CJ4Q7B 137653825 IC50 = 400 nM T16739 CU6SM3 137654538 IC50 = 210 nM T16739 C9T1SH 137654930 IC50 = 1200 nM T16739 C7H4YN 137655365 IC50 = 1600 nM T16739 CVI96M 137655554 IC50 = 245.8 nM T16739 CS23VK 137655643 IC50 = 4400 nM T16739 C76YWA 137655655 IC50 > 10000 nM T16739 CL0ST9 137655691 IC50 = 1153 nM T16739 CZ8FJ5 137655706 IC50 = 2633 nM T16739 CMKQ62 137655844 IC50 = 197.06 nM T16739 CLYZ81 137655983 IC50 = 1100 nM T16739 CH4PG0 137655999 IC50 > 10000 nM T16739 CKQ68E 137656309 IC50 > 150000 nM T16739 C8WE9Q 137656455 Ki = 60 nM T16739 C0OL6X 137656650 IC50 = 220 nM T16739 C7BQ1F 137656659 Ki > 500000 nM T16739 CK9ND3 137656985 Ki = 98 nM T16739 CTRE41 137657231 IC50 = 492.58 nM T16739 C24ELI 137657571 IC50 = 22700 nM T16739 CB45GJ 137657826 IC50 = 950 nM T16739 CCJG57 137657965 IC50 > 50000 nM T16739 CZXU25 137658111 IC50 = 190 nM T16739 C9WYS1 137658132 IC50 > 30000 nM T16739 CC15IZ 137658380 IC50 = 620 nM T16739 CLZ6F9 137658483 IC50 = 83 nM T16739 CT8KJ9 137658657 IC50 = 14200 nM T16739 CLGR74 137658796 IC50 > 10000 nM T16739 CIDO45 137658994 IC50 = 4200 nM T16739 C5PV0M 137659142 IC50 = 79 nM T16739 C76UYF 137659212 IC50 = 13900 nM T16739 C7C0WJ 137659602 IC50 = 1400 nM T16739 C2JXZ5 137659994 IC50 = 1190 nM T16739 C8QC4L 137660056 IC50 = 4300 nM T16739 CH9W5J 137660236 Ki > 500000 nM T16739 CHT3M9 137660431 IC50 = 6800 nM T16739 CE8Y5U 137660542 IC50 > 10000 nM T16739 C2HML9 137660640 IC50 = 154 nM T16739 CNV6O4 137660817 IC50 = 7500 nM T16739 CUZI37 137661062 IC50 > 10000 nM T16739 C0IGL6 137661623 IC50 > 10000 nM T16739 C2Z9JD 137661839 IC50 = 1000 nM T16739 C36GZV 137661855 IC50 = 121.23 nM T16739 CUP4N3 137662262 IC50 = 5500 nM T16739 C5AIQ9 138494685 IC50 = 15 nM T16739 CDHB24 138745757 EC50 = 140 nM T16739 C18VCF 141742824 IC50 = 4900 nM T16739 CWH5X3 145948592 IC50 = 17000 nM T16739 C97JVF 145948622 IC50 = 320 nM T16739 CU5N2J 145948654 IC50 = 40000 nM T16739 C9XO4M 145948655 IC50 = 280 nM T16739 C84JMU 145948688 IC50 = 63000 nM T16739 CHP2V5 145948690 IC50 = 8400 nM T16739 CLD12N 145949023 IC50 = 290 nM T16739 C5GM0U 145949030 IC50 = 440 nM T16739 CDA28I 145949712 IC50 = 1200 nM T16739 CO2M5E 145950303 IC50 = 490 nM T16739 CR34FK 145950671 IC50 = 21 nM T16739 C5DRL4 145951334 IC50 = 1990 nM T16739 C1E5VT 145951681 IC50 = 5950 nM T16739 CX1P7H 145952331 IC50 = 1300 nM T16739 CC4ET5 145952377 IC50 = 24900 nM T16739 CFH2D1 145953792 IC50 = 1090 nM T16739 CL0XT8 145954248 IC50 = 2210 nM T16739 C0TXG3 145954281 IC50 = 880 nM T16739 C37SYH 145955424 IC50 = 5000 nM T16739 CO5NR3 145955440 IC50 = 1870 nM T16739 C5XT4Z 145956132 IC50 = 17 nM T16739 CPY71F 145956290 EC50 = 3.6 nM T16739 CJ03TU 145957740 IC50 = 7160 nM T16739 C23WFS 145957776 IC50 = 8900 nM T16739 C1JKT0 145959891 IC50 = 76 nM T16739 CVP7Q0 145960268 IC50 > 30000 nM T16739 CRCO56 145963866 IC50 = 388.08 nM T16739 CI1UR7 145965143 IC50 = 881.51 nM T16739 CQ65IE 145965766 IC50 = 349.06 nM T16739 CC6ZF7 145965910 IC50 = 223.13 nM T16739 CID4J6 145966605 IC50 = 366.54 nM T16739 CP19XR 145966645 IC50 = 631.19 nM T16739 CW6UP9 145967077 IC50 = 828.31 nM T16739 CZOB60 145967223 IC50 = 26.13 nM T16739 CQV1S7 145969296 IC50 = 622 nM T16739 C34IVT 145971725 IC50 = 7300 nM T16739 C4GD2T 145971846 IC50 = 169.61 nM T16739 CM4FI9 145972729 IC50 = 423.42 nM T16739 CNE54W 145972804 IC50 = 154 nM T16739 C1WF7B 145973546 IC50 = 273.72 nM T16739 CNV7M2 145973643 IC50 = 221.97 nM T16739 CJSF01 145973737 IC50 = 147.7 nM T16739 CVN9B4 145973902 IC50 = 273.83 nM T16739 CY1G2F 145974565 IC50 = 3850 nM T16739 C1TI6B 145974586 IC50 = 180 nM T16739 C3L6BX 145975245 IC50 = 107 nM T16739 C9OM3Y 145975311 IC50 = 224.11 nM T16739 CZ24BU 145975518 IC50 = 350.26 nM T16739 CN9V7L 145976038 IC50 = 253.6 nM T16739 C6KDE9 145977476 IC50 = 110.25 nM T16739 C9M3KP 145977644 IC50 = 455.51 nM T16739 CIF4G8 145977849 IC50 = 201.23 nM T16739 CIXM06 145978256 IC50 = 91.83 nM T16739 CM71HX 145979766 IC50 = 122 nM T16739 CN6V4L 145979985 IC50 = 91.1 nM T16739 CUI5C2 145980623 IC50 = 51.8 nM T16739 CX4I9A 145980725 IC50 = 103.9 nM T16739 C91YZF 145980909 IC50 = 114.1 nM T16739 CW41TN 145981088 IC50 = 325 nM T16739 CVT4N5 145981092 IC50 = 117 nM T16739 CK0V8L 145981246 IC50 = 146.5 nM T16739 C8EQ1I 145981399 IC50 = 643.5 nM T16739 CL23TD 145981420 IC50 = 79.7 nM T16739 CT82OJ 145981451 IC50 = 82.6 nM T16739 C5XTS3 145982234 IC50 = 154.5 nM T16739 CG34HN 145983490 IC50 = 410 nM T16739 CDK5E3 145983937 IC50 = 64.5 nM T16739 CD9XT8 145984039 IC50 = 1200 nM T16739 C7U8QY 145984922 IC50 = 157.9 nM T16739 C2KY9O 145985822 IC50 > 75000 nM T16739 CRGD07 145985886 IC50 = 4400 nM T16739 C7MBT5 145986835 IC50 = 111.7 nM T16739 CW3RG1 145987055 IC50 = 77.5 nM T16739 C7UGL8 145987433 IC50 = 159 nM T16739 CE4CW1 145987550 IC50 = 202.8 nM T16739 C2Q5UT 145987662 IC50 = 417.5 nM T16739 C2R9GZ 145987759 IC50 = 294.5 nM T16739 C0JTV3 145988106 IC50 = 69.1 nM T16739 C0VRL2 145988393 IC50 = 187.3 nM T16739 CX5F4Z 145989197 IC50 = 60 nM T16739 C2PZ1M 145989589 IC50 = 90 nM T16739 CS5G2V 145989627 IC50 = 202.4 nM T16739 CJFG45 145990271 IC50 = 91 nM T16739 C7GLE9 145990404 IC50 = 110 nM T16739 C2K7VD 145990489 IC50 = 276.5 nM T16739 CPQK41 145990550 IC50 = 112.1 nM T16739 C87IWX 145990849 IC50 = 100 nM T16739 C1L9RX 145991036 IC50 = 817.1 nM T16739 CI0X6F 145991237 IC50 = 80.7 nM T16739 C4HOG1 145991279 IC50 = 35.3 nM T16739 CTH12U 145991708 IC50 = 119.9 nM T16739 C9PVF0 145991993 IC50 = 94.9 nM T16739 C54FDN 145992291 IC50 = 66.5 nM T16739 CWS5K0 145992436 IC50 = 117.5 nM T16739 CM0DW5 145993841 IC50 = 194.6 nM T16739 CK58BJ 145994205 IC50 = 108.5 nM T16739 C5OJV6 145994210 IC50 = 95.9 nM T16739 CGD7X6 149035905 IC50 > 10000 nM T16739 CH82YB 149430327 IC50 > 10000 nM T16739 CL9I0N 153241388 IC50 > 10000 nM T16739 C1VRF0 155511266 IC50 > 100000 nM T16739 CXS8C7 155511320 IC50 > 50000 nM T16739 C14FHM 155512092 IC50 = 283 nM T16739 CY4W6M 155512249 IC50 = 1.4 nM T16739 C8Z3MI 155512516 IC50 > 100000 nM T16739 C54NIK 155512517 IC50 = 124.05 nM T16739 CK8AH7 155512564 IC50 > 100000 nM T16739 CJ08BN 155513545 IC50 = 17620 nM T16739 C1I7MX 155513834 IC50 = 8410 nM T16739 CK5L7C 155514006 IC50 > 10000 nM T16739 C63TMW 155514054 IC50 > 100000 nM T16739 CTQ3F4 155514293 IC50 = 240.5 nM T16739 CE2CB7 155514322 IC50 = 8600 nM T16739 COFQ57 155514340 IC50 = 2960 nM T16739 CWL09M 155514551 IC50 = 6160 nM T16739 C3MCO5 155514879 IC50 = 17380 nM T16739 CQ9C4H 155515673 IC50 > 50000 nM T16739 C3JM6E 155515729 IC50 = 32560 nM T16739 CJ03RP 155515798 IC50 = 88300 nM T16739 C1F6GM 155515963 IC50 = 211.35 nM T16739 CU57MI 155515979 IC50 > 10000 nM T16739 C0AEO1 155516202 IC50 > 50000 nM T16739 C89HFY 155516699 IC50 = 31350 nM T16739 CA8E3D 155516736 IC50 = 8130 nM T16739 CTYB35 155516772 IC50 > 10000 nM T16739 C3C4EB 155516903 IC50 = 6200 nM T16739 C6AOU3 155516972 IC50 = 9030 nM T16739 CB6V9A 155517388 IC50 > 100000 nM T16739 CQ09GC 155517887 IC50 = 9469 nM T16739 CO8NF7 155518169 IC50 = 11780 nM T16739 CIQ3H5 155518602 IC50 = 20497 nM T16739 C36LGV 155519027 IC50 = 187 nM T16739 CX4AT1 155519230 IC50 = 12390 nM T16739 C2NAH8 155519577 IC50 > 10000 nM T16739 C10FOR 155519973 IC50 = 80670 nM T16739 C74KVA 155520222 IC50 > 100000 nM T16739 CJZ8O0 155520641 IC50 > 100000 nM T16739 CY0AE8 155521035 IC50 = 21200 nM T16739 CUT0R6 155521354 IC50 = 11500 nM T16739 CZT80M 155521515 IC50 = 1400 nM T16739 C9JS2I 155522001 IC50 > 50000 nM T16739 C5AGQ0 155522019 IC50 > 10000 nM T16739 C4YPF9 155522024 IC50 = 364 nM T16739 CZ1BA4 155522435 IC50 = 1800 nM T16739 CTM76G 155522838 IC50 = 14840 nM T16739 C5N2GX 155523580 IC50 > 10000 nM T16739 CA4GF8 155524054 IC50 = 25130 nM T16739 CHL60A 155524060 IC50 = 5800 nM T16739 CV6LQ2 155524438 IC50 = 5903 nM T16739 C1H4ZM 155524754 IC50 = 25780 nM T16739 C2PCF7 155524926 IC50 = 2320 nM T16739 C0N6YU 155525438 IC50 > 10000 nM T16739 CZK1F8 155525945 IC50 > 100000 nM T16739 C8N0QO 155526083 IC50 = 8210 nM T16739 C2S0CL 155526249 IC50 = 38130 nM T16739 C4NQF1 155526272 IC50 > 100000 nM T16739 C93DAF 155526361 IC50 = 16170 nM T16739 COC04K 155526480 IC50 = 28130 nM T16739 C1KS8M 155526964 IC50 > 10000 nM T16739 CQ6S4V 155527134 IC50 > 100000 nM T16739 CZ4V2P 155527186 IC50 = 23090 nM T16739 C8XIB0 155527448 IC50 = 2600 nM T16739 CTK4B6 155527517 IC50 > 10000 nM T16739 CKH5S7 155527758 IC50 > 10000 nM T16739 CO9K7S 155527956 IC50 > 10000 nM T16739 CJXU81 155527961 IC50 > 100000 nM T16739 C39ZEQ 155528113 IC50 = 4000 nM T16739 CXR62G 155528241 IC50 > 100000 nM T16739 CCA76W 155528448 IC50 = 301 nM T16739 C1W9RV 155528515 IC50 > 10000 nM T16739 CE2J7B 155528539 IC50 > 100000 nM T16739 C4JB9V 155528847 IC50 > 100000 nM T16739 C7IQB3 155528938 IC50 = 1400 nM T16739 CM86DU 155528956 IC50 > 100000 nM T16739 CQM2L6 155529262 IC50 = 720 nM T16739 C6ZR3K 155529304 IC50 > 100000 nM T16739 C2Y5JU 155529473 IC50 > 100000 nM T16739 C0I7CO 155529614 IC50 > 10000 nM T16739 CZ39JY 155529671 IC50 = 8890 nM T16739 CKP95A 155529723 IC50 = 14250 nM T16739 C84LQC 155529930 IC50 > 100000 nM T16739 C0H3AR 155529958 IC50 = 6200 nM T16739 CJO4L9 155530140 IC50 > 100000 nM T16739 CJK4V9 155530484 IC50 > 100000 nM T16739 CR7K1U 155531166 IC50 = 19850 nM T16739 CM9PE3 155531622 IC50 > 10000 nM T16739 C5A8MO 155532280 IC50 = 14200 nM T16739 CGI2K5 155532419 IC50 > 10000 nM T16739 CMKP85 155532627 IC50 = 800 nM T16739 C9RJ7Y 155532890 IC50 > 10000 nM T16739 CZQ6I5 155533215 IC50 > 10000 nM T16739 CF3Y9J 155533893 IC50 = 15340 nM T16739 CIGO02 155534062 IC50 = 22520 nM T16739 CCQ16F 155534151 IC50 = 10300 nM T16739 CE1I2D 155534448 IC50 = 1784 nM T16739 C1TVH7 155534458 IC50 > 10000 nM T16739 CR47VA 155534676 IC50 = 49600 nM T16739 C7QT8G 155535122 IC50 > 100000 nM T16739 CV1RP6 155535358 IC50 > 100000 nM T16739 C6C8RT 155535388 IC50 > 10000 nM T16739 CE53GM 155535765 IC50 > 10000 nM T16739 C0HZN9 155536909 IC50 > 50000 nM T16739 C9AQ3H 155536932 IC50 > 50000 nM T16739 C7RM1Z 155537544 IC50 > 50000 nM T16739 CBH32R 155537569 IC50 = 4240 nM T16739 CX94TW 155537667 IC50 = 1720 nM T16739 C34MHK 155537841 IC50 > 50000 nM T16739 C48ZJF 155537966 IC50 > 100000 nM T16739 C94GAK 155538209 IC50 > 10000 nM T16739 C0ZRK2 155538344 IC50 = 9550 nM T16739 CU98MX 155538436 IC50 > 50000 nM T16739 C0SZR7 155538813 IC50 > 50000 nM T16739 C5IL8M 155540041 IC50 = 764 nM T16739 CQR25J 155540292 IC50 > 50000 nM T16739 C2K9MT 155540654 IC50 > 10000 nM T16739 CIS43T 155540722 IC50 > 50000 nM T16739 C2OH4K 155541274 IC50 = 29240 nM T16739 CSA8Z2 155541837 IC50 > 50000 nM T16739 C6M9XC 155541996 IC50 = 3570 nM T16739 CX4P8S 155542351 IC50 = 109.35 nM T16739 C7I8TH 155542625 IC50 = 4500 nM T16739 CH9I1F 155542865 IC50 > 100000 nM T16739 CHTB05 155543040 IC50 > 50000 nM T16739 CS68OT 155543573 IC50 = 2.3 nM T16739 CIGP59 155544097 IC50 > 50000 nM T16739 CB1XH5 155544104 IC50 = 692.15 nM T16739 CUZ6H8 155544121 IC50 = 5130 nM T16739 CV5OL7 155544292 IC50 = 8959 nM T16739 CLUK20 155544445 IC50 > 10000 nM T16739 C8IB7D 155544714 IC50 > 100000 nM T16739 C2H1WQ 155544893 IC50 = 21150 nM T16739 CD7E9T 155545053 IC50 = 24420 nM T16739 CGWL63 155545059 IC50 > 100000 nM T16739 CTQR16 155545374 IC50 = 25750 nM T16739 CMPJ65 155545619 IC50 = 1610 nM T16739 C8OCU5 155546210 IC50 = 12410 nM T16739 C2WCH1 155546411 IC50 = 18510 nM T16739 C60OKG 155547117 IC50 = 66.13 nM T16739 COMN19 155547339 IC50 = 5900 nM T16739 CU5FK4 155548497 IC50 > 10000 nM T16739 CD0BN9 155548800 IC50 > 10000 nM T16739 CJP91E 155549020 IC50 > 10000 nM T16739 CU78SJ 155549223 IC50 > 10000 nM T16739 C9SXF1 155549673 IC50 = 13120 nM T16739 CCE7I0 155549909 IC50 > 50000 nM T16739 C12BVP 155550124 IC50 = 28430 nM T16739 CE8UN2 155550382 IC50 > 100000 nM T16739 CT96SQ 155550749 IC50 > 100000 nM T16739 C6H1BC 155550901 IC50 = 18960 nM T16739 C32TCH 155551024 IC50 > 10000 nM T16739 C5YH3M 155551273 IC50 = 20850 nM T16739 CM3VB6 155551391 IC50 = 6000 nM T16739 C6FPC5 155551554 IC50 > 100000 nM T16739 CMU06X 155551632 IC50 > 10000 nM T16739 C8JD0O 155551671 IC50 = 61.04 nM T16739 C45JYO 155551739 IC50 > 10000 nM T16739 CW4O3P 155551783 IC50 > 50000 nM T16739 CH3O7Y 155552967 IC50 = 5849 nM T16739 C3KBT2 155552984 IC50 > 100000 nM T16739 C78CAG 155553021 IC50 > 100000 nM T16739 C82NZQ 155553274 IC50 = 4.6 nM T16739 CQ5NF1 155553305 IC50 = 4467 nM T16739 C48XOL 155553511 IC50 = 2900 nM T16739 CXK90C 155553926 IC50 > 100000 nM T16739 CO3VZ7 155554343 IC50 > 100000 nM T16739 CBQL25 155554680 IC50 > 100000 nM T16739 CT6Y1L 155554736 IC50 > 10000 nM T16739 CWFU34 155554942 IC50 > 50000 nM T16739 CQKH19 155555069 IC50 = 184.15 nM T16739 CC02EV 155555071 IC50 = 1230 nM T16739 C6YF2A 155555194 IC50 = 53000 nM T16739 CR5NI3 155555689 IC50 > 10000 nM T16739 C1GE8S 155555798 IC50 = 1470 nM T16739 C3B9FR 155556977 IC50 > 10000 nM T16739 CTVQ18 155557424 IC50 = 359.7 nM T16739 C1E3KJ 155557461 IC50 > 100000 nM T16739 C3S6KC 155557528 IC50 = 25810 nM T16739 CYRD91 155557589 IC50 > 50000 nM T16739 CM7C9S 155557939 IC50 > 10000 nM T16739 CSR8O1 155557945 IC50 = 12100 nM T16739 CO1R6S 155558109 IC50 > 100000 nM T16739 C3LHI6 155560394 IC50 > 50000 nM T16739 CDA1M9 155560663 IC50 > 100000 nM T16739 C2Z0FO 155560802 IC50 > 10000 nM T16739 CR8DS5 155560849 IC50 > 100000 nM T16739 C09JMY 155561128 IC50 = 920 nM T16739 CI9BP6 155561362 IC50 > 50000 nM T16739 CY21GB 155561565 IC50 = 33900 nM T16739 CU9Y7O 155561599 IC50 = 8980 nM T16739 C5R3LT 155561606 IC50 = 84.38 nM T16739 C2JQ3C 155561938 IC50 = 2800 nM T16739 C9N4FD 155561982 IC50 > 50000 nM T16739 C8I6TY 155562066 IC50 = 1290 nM T16739 CN07GK 155562384 IC50 > 50000 nM T16739 CU79CI 155562928 IC50 > 100000 nM T16739 CR3N4L 155563005 IC50 > 10000 nM T16739 C9EQS8 155563020 IC50 = 859 nM T16739 COIA41 155563202 IC50 = 5870 nM T16739 C9QV7A 155563234 IC50 = 30140 nM T16739 CEY9G4 155563653 IC50 > 100000 nM T16739 CWYL58 155563836 IC50 > 100000 nM T16739 CLN70O 155564275 IC50 > 50000 nM T16739 CS0UY1 155564350 IC50 = 19350 nM T16739 C6GUF2 155564945 IC50 = 22860 nM T16739 C29SXL 155564963 IC50 = 11210 nM T16739 CI2W5M 155565400 IC50 > 50000 nM T16739 CRKI14 155565934 IC50 > 50000 nM T16739 C83QKU 155566043 IC50 > 10000 nM T16739 C2B9KQ 155566623 IC50 > 10000 nM T16739 C8UPR7 155566682 IC50 > 50000 nM T16739 CC4Q2I 155567001 IC50 > 10000 nM T16739 CX0W5G 155567229 IC50 = 4.9 nM T16739 CVK5F7 155567996 IC50 = 7800 nM T16739 CUQX17 155568039 IC50 > 100000 nM T16739 C1J4PU 155568294 IC50 = 25740 nM T16739 CX1GM4 155568297 IC50 > 100000 nM T16739 CI8O0Q 155568425 IC50 = 6580 nM T16739 CA0E8D 155568764 IC50 > 10000 nM T16739 C6D4WP 155568813 IC50 = 15630 nM T16739 C8S0FZ 155568919 IC50 = 252.33 nM T16739 CFAX90 155569105 IC50 = 8344 nM T16739 CJMN49 155569426 IC50 > 10000 nM T16739 C4TD6A 155569455 IC50 > 50000 nM T16739 CQ49MC 155569602 IC50 > 100000 nM T16739 C50XIE 155569635 IC50 > 100000 nM T16739 D00MXS 5281703 IC50 = 8870 nM T16739 D00RFY 5281612 IC50 = 27900 nM T16739 D00YEV 5281605 IC50 = 12500 nM T16739 D03LGV 11241513 IC50 = 6700 nM T16739 D06TLQ 5488822 IC50 = 16700 nM T16739 D08PHY 11171752 IC50 > 25000 nM T16739 D09ALJ 5280805 IC50 = 2160 nM T16739 D09HBX 10374615 IC50 > 25000 nM T16739 D0C8SX 56639570 IC50 = 20 nM T16739 D0EV7U 71522234 IC50 = 24 nM T16739 D0F2DC 11816512 IC50 > 25000 nM T16739 D0H1VT 11423691 IC50 > 25000 nM T10383 D01XBA 5035 IC50 = 3400 nM T10383 D03JRG 46937439 IC50 = 20 nM T10383 D0CI4A 25105704 IC50 = 380 nM T10383 D0OX9E 50902705 IC50 = 700 nM T10383 CQ0IC4 63062 IC50 = 44 nM T10383 CW21VY 16739265 IC50 = 300 nM T10383 C17GSK 21428808 IC50 = 610 nM T10383 C89GXW 21428832 IC50 = 1410 nM T10383 C3IHB0 21428850 IC50 = 130 nM T10383 C9QY5H 21428857 IC50 = 1400 nM T10383 CBS6E1 21428871 IC50 = 1500 nM T10383 CVC98H 21428895 IC50 = 76 nM T10383 C23HQA 21428932 IC50 = 5670 nM T10383 C40CFO 21428968 IC50 = 8000 nM T10383 CK90LC 21428971 IC50 = 1100 nM T10383 C8IXU1 21429000 IC50 = 240 nM T10383 CT0C3Z 25105692 IC50 = 210 nM T10383 CA7XR1 25105696 IC50 > 2000 nM T10383 CRG7X8 25105698 IC50 = 130 nM T10383 C54TAV 25105699 IC50 = 220 nM T10383 CIPH75 25105700 IC50 = 1100 nM T10383 C9H5WS 25105701 IC50 = 210 nM T10383 CMJ14L 25105702 IC50 = 1400 nM T10383 C7EW5O 25105703 IC50 = 79 nM T10383 C9J7ZI 25105705 IC50 = 600 nM T10383 CMW3Y1 25105706 IC50 = 3900 nM T10383 C5MZX7 25105707 IC50 = 1000 nM T10383 C2ZF1U 25105708 IC50 > 20000 nM T10383 C68JBL 25105709 IC50 = 340 nM T10383 CF6P7E 25105710 IC50 = 170 nM T10383 C30IGQ 25105711 IC50 = 2200 nM T10383 C19VQY 25105712 IC50 = 12000 nM T10383 C9TX2Y 25105713 IC50 = 1800 nM T10383 C48BVE 25105714 IC50 = 4300 nM T10383 C3WPU2 25105715 IC50 = 110 nM T10383 C8XHA1 25105716 IC50 = 1200 nM T10383 CH2A5B 44138051 IC50 = 140 nM T10383 CU5D9O 44438308 IC50 = 1000 nM T10383 CO0V5A 44438309 IC50 = 42 nM T10383 C3DW6Q 44438310 IC50 = 20 nM T10383 CXB2R1 44573118 IC50 = 1200 nM T10383 CT6FP3 44573119 IC50 = 1150 nM T10383 COD46G 44573120 IC50 = 730 nM T10383 C65LXN 44573121 IC50 = 187 nM T10383 CD6G3I 44573130 IC50 = 890 nM T10383 C40TOA 44573131 IC50 = 6400 nM T10383 CRC8G1 44573132 IC50 = 360 nM T10383 C8N3CM 44573176 IC50 = 3900 nM T10383 C0D4GS 44573191 IC50 = 3800 nM T10383 CSZ0W7 44573597 IC50 = 730 nM T10383 CFQA45 44573598 IC50 = 740 nM T10383 C8Q5RD 44573599 IC50 = 860 nM T10383 CC09AZ 44573641 IC50 = 850 nM T10383 C39HWT 44573687 IC50 = 140 nM T10383 CT18AS 44573688 IC50 = 61 nM T10383 CWI75L 44573689 IC50 = 375 nM T10383 C14ZEX 44573690 IC50 = 97 nM T10383 C8A4LR 44573727 IC50 = 42 nM T10383 CBM42C 44573728 IC50 = 14 nM T10383 CBCX36 44573767 IC50 = 12000 nM T10383 C5BDG2 44573768 IC50 = 10000 nM T10383 CQ9X2N 44573769 IC50 = 14000 nM T10383 CQ62KR 44573770 IC50 = 13000 nM T10383 CB2G5X 44573806 IC50 > 20000 nM T10383 C1GM3U 44573807 IC50 = 3100 nM T10383 CZO1C6 44573808 IC50 = 1040 nM T10383 CEX9F5 44573809 IC50 = 1400 nM T10383 CP63HT 44591888 IC50 > 20000 nM T10383 CK8GV2 44591889 IC50 = 90 nM T10383 CHVO21 44591890 IC50 = 1600 nM T10383 CP5VO4 44591891 IC50 = 30000 nM T10383 C09BTI 44591892 IC50 = 200 nM T10383 C9E5ZV 44591930 IC50 = 30 nM T10383 CCX35M 44591931 IC50 = 990 nM T10383 CDY58B 44591932 IC50 = 550 nM T10383 CBHW79 44591933 IC50 > 20000 nM T10383 CFOX18 44591934 IC50 = 27000 nM T10383 C0J3UF 46938432 IC50 = 25 nM T10383 C8LAD0 46938434 IC50 = 73 nM T10383 CMB63C 46938535 IC50 = 100 nM T10383 C3GPY4 46938537 IC50 = 30 nM T10383 CNSZ76 46938539 IC50 = 50 nM T10383 CRN3Z8 46938541 IC50 = 100 nM T10383 CYO78K 46938928 IC50 = 60 nM T10383 CB06NU 46939226 IC50 = 63 nM T10383 CP04XW 46939227 IC50 = 350 nM T10383 C4B2SF 46939228 IC50 = 290 nM T10383 CV8DS2 46939229 IC50 = 165 nM T10383 CX3QE6 46939321 IC50 = 70 nM T10383 C2K4TB 46939322 IC50 = 120 nM T10383 CR7L9X 46939323 IC50 = 70 nM T10383 CQI17K 46939324 IC50 = 660 nM T10383 CJ7VN8 46939407 IC50 = 80 nM T10383 C2ZW8V 46939408 IC50 = 40 nM T10383 CO5X0P 46939409 IC50 = 655 nM T10383 CY05QU 46939410 IC50 = 200 nM T10383 C1PZM4 46939489 IC50 = 350 nM T10383 CX49SE 46939490 IC50 = 360 nM T10383 C14XNH 49850293 IC50 = 140 nM T10383 CF31UA 50902617 IC50 = 2800 nM T10383 C58APV 50902621 IC50 = 4000 nM T10383 CPUG80 50902623 IC50 = 220 nM T10383 C3RNG4 50902707 IC50 = 810 nM T10383 CH38VC 50902709 IC50 = 3175 nM T10383 CRC6V8 50902786 IC50 = 450 nM T10383 C16FQK 50902788 IC50 = 43 nM T10383 CKE14R 50902876 IC50 = 60 nM T10383 CAJ3L1 50902978 IC50 = 12 nM T10383 C47VGW 53393916 IC50 = 355 nM T10383 C26TVP 56593045 IC50 = 120 nM T10383 CB27OD 56593054 IC50 = 20 nM T10383 C2XP8D 56593056 IC50 = 200 nM T10383 C3ZYA2 56593082 IC50 = 35 nM T10383 C7ENU3 56846622 IC50 = 3450 nM T10383 C1CBU4 56846623 IC50 = 1060 nM T10383 CEZA46 56846640 IC50 = 800 nM T10383 C47LNP 68182778 IC50 = 210 nM T10383 CBME89 68182839 IC50 = 26 nM T10383 C6AHP7 68183060 IC50 = 150 nM T10383 COXN56 68188986 IC50 = 115 nM T10383 CUBM27 71716675 IC50 = 520 nM T10383 CWB3V1 71718136 IC50 = 20 nM T10383 CRG3Z8 73099418 IC50 = 360 nM T10383 C92QNG 155537801 IC50 = 2.5 nM T10383 CVU9P7 155540036 IC50 = 70 nM T10383 D07RPV 65490 IC50 = 310 nM T77548 D00ENY 33032 IC50 = 5.7 nM T77548 D0B6RA 9834591 EC50 = 47773 nM T77548 D0D4OW 57338826 IC50 = 1900 nM T77548 D0U5CS 213056 EC50 = 11470 nM T77548 D0ZV0R 16660135 IC50 > 10000 nM T77548 CB15YI 125799 EC50 > 300000 nM T77548 CO9KU6 443586 Ki > 1000000 nM T77548 COJV81 4521898 EC50 > 10000 nM T77548 C05WNA 5310956 Ki = 3400 nM T77548 C3RTI9 6348408 EC50 = 6500 nM T77548 C9PJQ1 9794208 EC50 = 6530 nM T77548 C9XQK6 10198133 EC50 = 7340 nM T77548 CMW4B2 10353365 EC50 = 3070 nM T77548 CZ09YG 10358265 IC50 > 300000 nM T77548 CQ1L0O 10359073 Ki > 300000 nM T77548 CYL91R 10456810 IC50 = 990 nM T77548 CDO7A1 10979251 EC50 > 25000 nM T77548 CJ5B8P 11084869 EC50 > 25000 nM T77548 C8LSU6 11275666 EC50 > 25000 nM T77548 CL1VX3 11310142 EC50 > 25000 nM T77548 CX2T1N 11344646 EC50 > 25000 nM T77548 CSW38G 15420544 EC50 > 10000 nM T77548 CP9Y7Q 15479143 EC50 = 11500 nM T77548 CJS57V 16061421 EC50 = 300 nM T77548 C6Q4GL 16747847 EC50 = 340 nM T77548 CM7JD0 16747848 EC50 = 2150 nM T77548 CWU3X9 16748099 EC50 = 6510 nM T77548 CS5B7A 18138918 IC50 > 30000 nM T77548 C0K9DR 22884216 IC50 > 1000000 nM T77548 CI9FL7 24779948 EC50 = 125000 nM T77548 CJR05E 24780088 EC50 = 141000 nM T77548 CW3S6A 24780089 EC50 = 511000 nM T77548 CQ1S9T 24780091 EC50 = 34000 nM T77548 C5OQ7F 24780092 EC50 > 100000 nM T77548 C7F4YL 24780225 EC50 = 7600 nM T77548 CNF72Q 44190035 IC50 > 10000 nM T77548 CL13FV 44302605 IC50 > 300000 nM T77548 C03QML 44302608 IC50 > 300000 nM T77548 C2H6QV 44302609 IC50 > 300000 nM T77548 CP1QS5 44302686 IC50 > 300000 nM T77548 C0V9DN 44302818 IC50 > 300000 nM T77548 CDM1P2 44302819 IC50 > 300000 nM T77548 C1GV9Q 44302837 IC50 > 300000 nM T77548 C34AVQ 44302856 IC50 > 300000 nM T77548 CWV7F0 44322840 Ki = 15000 nM T77548 CR1OL6 44328753 IC50 = 490 nM T77548 CUA80G 44328850 IC50 = 1230 nM T77548 C2SH0O 44329024 IC50 = 2250 nM T77548 CX0Y4F 44329029 IC50 = 5180 nM T77548 C76LOU 44329031 IC50 = 750 nM T77548 CCV4N5 44329032 IC50 = 340 nM T77548 CDP86T 44329033 IC50 = 380 nM T77548 C9V5XC 44329042 IC50 = 2520 nM T77548 CKB74O 46918013 EC50 = 1200 nM T77548 C1VY4Z 46918015 EC50 = 42000 nM T77548 C7KSH2 46918017 EC50 = 20000 nM T77548 CE4KP1 51050257 Ki > 10000 nM T77548 CN1HU8 53235518 EC50 > 10000 nM T77548 CY58NO 53240406 EC50 = 10100 nM T77548 CW36CH 53322382 EC50 > 10000 nM T77548 CIHC67 54582001 IC50 > 30000 nM T77548 CZ0A1T 57765525 EC50 = 1600 nM T77548 CE7DU0 57765529 EC50 = 4600 nM T77548 C6N0PK 57765531 EC50 = 2700 nM T77548 C49IAZ 57765535 EC50 = 2500 nM T77548 C4BZ0U 57765536 EC50 = 490 nM T77548 C9QDZ0 57765549 EC50 > 100000 nM T77548 C90MQS 57765556 EC50 = 4500 nM T77548 CHQM83 57765572 EC50 = 5200 nM T77548 C4T6JE 57765594 EC50 = 4200 nM T77548 C1K5DT 57765607 EC50 = 21200 nM T77548 CSI9E0 57765613 EC50 = 660 nM T77548 CZ4KT6 57765615 EC50 = 2900 nM T77548 CBFD61 57765616 EC50 = 980 nM T77548 CC82HD 57765622 EC50 = 1540 nM T77548 CQ70WE 57765633 EC50 = 1900 nM T77548 CISA81 58058356 EC50 = 5400 nM T77548 CPDW56 58058372 EC50 = 1000 nM T77548 CQY10C 58058380 EC50 = 33000 nM T77548 CY2NR8 58058384 EC50 = 2200 nM T77548 C8JAU2 60096211 EC50 = 4300 nM T77548 C8N4UB 60096231 EC50 > 25000 nM T77548 CBX67G 67246999 EC50 > 10000 nM T77548 C5K7QG 67974411 EC50 > 10000 nM T77548 C0BC6D 68012045 EC50 = 28000 nM T77548 CCT07V 68290289 EC50 > 10000 nM T77548 C03JUE 68290572 EC50 > 10000 nM T77548 CG7F5Z 70051296 EC50 > 25000 nM T77548 CBK2Y6 70051926 EC50 = 1590 nM T77548 CZ6XT7 70052526 EC50 > 25000 nM T77548 C8U0CT 71681823 EC50 = 12400 nM T77548 CO5P1V 71681824 EC50 > 25000 nM T77548 C6EIO9 71681825 EC50 = 12000 nM T77548 CLH9N3 71681826 EC50 > 25000 nM T77548 CXW8R2 72714783 EC50 > 10000 nM T77548 C07OAB 87618914 EC50 = 6600 nM T77548 C0VN8X 92044496 EC50 = 380 nM T77548 CUC13P 122187795 IC50 > 30000 nM T77548 CCP5U2 122195692 EC50 > 10000 nM T77548 CH2AO4 122539788 IC50 > 30000 nM T77548 C2MEI0 124425164 EC50 = 26000 nM T77548 CFC05Q 131954513 EC50 = 2600 nM T77548 C3EGM5 137321168 IC50 > 10000 nM T77548 C0M7EV 137631886 EC50 = 26200 nM T77548 CI4V1F 137631983 EC50 = 14000 nM T77548 C8QU9Z 137632643 EC50 = 6500 nM T77548 C4E7KH 137634091 EC50 = 25000 nM T77548 C2WJ3T 137634489 EC50 = 29700 nM T77548 CS7O0A 137634883 EC50 = 2500 nM T77548 CQ02YR 137635378 EC50 = 6900 nM T77548 CTG5M8 137635566 EC50 = 22800 nM T77548 CU2JA5 137636549 EC50 = 17000 nM T77548 C0KAJ3 137638200 EC50 = 38000 nM T77548 C9A8MG 137638288 EC50 = 22000 nM T77548 C9H6NY 137639752 EC50 = 31400 nM T77548 CK2W6L 137640190 EC50 = 1250 nM T77548 C7KT0R 137642290 EC50 = 19800 nM T77548 CAI63F 137642874 EC50 = 1300 nM T77548 CJHL32 137643079 EC50 = 219000 nM T77548 CNY07D 137643617 EC50 = 7200 nM T77548 C1FCY7 137643759 EC50 = 8400 nM T77548 CS5F0B 137644345 EC50 = 61000 nM T77548 C9U6EI 137645989 EC50 = 18000 nM T77548 CCW58E 137646034 EC50 = 277000 nM T77548 C3PDO0 137647077 EC50 = 2200 nM T77548 CEBV64 137649482 EC50 = 1800 nM T77548 CUH06J 137649749 EC50 = 9200 nM T77548 CO9L1G 137650519 EC50 = 23400 nM T77548 CQKZ08 137651515 EC50 = 40000 nM T77548 CYK1P7 137651881 EC50 = 81000 nM T77548 C6CW1G 137652072 EC50 = 36000 nM T77548 CT1M7B 137654697 EC50 = 39800 nM T77548 CMQ61F 137655963 EC50 = 17100 nM T77548 C5OK1E 137659207 EC50 = 35400 nM T77548 CDWR37 137661492 EC50 = 28000 nM T77548 C9C8KU 137661528 EC50 = 34300 nM T77548 CWA8H2 145955288 EC50 = 2900 nM T77548 C76FVC 155518354 EC50 = 890 nM T77548 CYXE53 155538270 IC50 > 10000 nM T77548 D00EPM 73755217 IC50 > 30000 nM T77548 D00IGI 2207 IC50 = 5.1 nM T77548 D01EVA 6278000 Ki > 100000 nM T77548 D04DKM 104766 Ki = 45000 nM T77548 D05TFE 5218788 Ki > 100000 nM T77548 D06PAK 10058694 Ki = 7300 nM T77548 D07GRG 10197984 EC50 = 1690 nM T77548 D09AQK 4545574 Ki = 210 nM T77548 D09QUN 58368068 EC50 > 10000 nM T77548 D09RPR 16737207 Ki > 10000 nM T77548 D0EK6P 5310984 Ki > 100000 nM T77548 D0IO8J 3025961 Ki > 100000 nM T77548 D0KL4K 71041983 EC50 = 29200 nM T77548 D0LC5O 16062593 EC50 = 23 nM T77548 D0N0NJ 15508178 IC50 > 300000 nM T77548 D0N2TP 44190040 IC50 > 10000 nM T77548 D0N9UZ 9819927 Ki = 170 nM T77548 D0OS8Y 15985251 IC50 > 10000 nM T77548 D0OV2V 6324634 Ki > 300000 nM T77548 D0PN6Z 179394 EC50 = 60 nM T77548 D0Q6VH 5311432 Ki > 100000 nM T77548 D0W3PY 6604820 EC50 = 5100 nM T38134 D0E3TC 44259 IC50 = 42 nM T38134 C38FDZ 16760660 IC50 = 0.12 ug.mL-1 T38134 C3VRO9 44557921 IC50 > 10000 nM T38134 CV63UL 67240318 IC50 > 10000 nM T38134 C2AN7T 134611886 IC50 > 100000 nM T38134 C2MD1Q 155513187 IC50 > 10000 nM T82078 CKA2Q3 8030846 EC50 = 560 nM T82078 CV71BY 11491636 IC50 = 230 nM T82078 C09ZEH 11600631 IC50 = 5000 nM T82078 COW07X 11643706 IC50 = 900 nM T82078 CLW30D 13633114 EC50 = 6430 nM T82078 C7JVW2 25157439 IC50 = 460 nM T82078 C1DSU6 44405462 IC50 = 950 nM T82078 C8VJ5F 44405524 IC50 = 1250 nM T82078 CF5WB8 44405603 IC50 = 2150 nM T82078 CBH7W9 44405604 IC50 = 5200 nM T82078 CA0GC9 44405661 IC50 = 22000 nM T82078 C12EAM 44405768 IC50 = 6460 nM T82078 C0Q5XC 44405780 IC50 = 6900 nM T82078 CBZ97N 44405822 IC50 = 1600 nM T82078 CN23KH 44589027 IC50 = 240 nM T82078 CBNO65 44589028 IC50 = 900 nM T82078 CHG12U 46201898 IC50 = 1200 nM T82078 C7X3PH 46205782 IC50 = 48 nM T82078 CDG83H 46732368 EC50 = 350 nM T82078 C9SFC7 46732463 EC50 = 8550 nM T82078 CBE2P6 54679465 EC50 = 300 nM T82078 C3W4DU 56655503 EC50 = 0.26 nM T82078 CB3AF0 56849710 EC50 = 0.45 nM T82078 CWC72K 56849711 EC50 = 1 nM T82078 CU7Q1J 56849712 EC50 = 0.87 nM T82078 C9TX4L 56849854 EC50 > 1000 nM T82078 C37INL 56849985 EC50 = 6.48 nM T82078 CSAM54 56849987 EC50 = 0.56 nM T82078 CG3IS5 56850128 EC50 = 1.47 nM T82078 C8X4NH 56850131 EC50 > 1000 nM T82078 CT1J9P 56850266 EC50 = 2.11 nM T82078 C3GCL2 56850401 EC50 = 1.55 nM T82078 CV0HU7 56850403 EC50 = 3.23 nM T82078 CX95CN 56850406 EC50 = 1.95 nM T82078 C3UHQ9 56850535 EC50 = 1.86 nM T82078 CW4ZC5 56850682 EC50 = 3.63 nM T82078 CSHE59 56850818 EC50 > 1000 nM T82078 C25HAU 56850822 EC50 > 1000 nM T82078 CUAK61 56850940 EC50 > 1000 nM T82078 CQJ4W0 56851062 EC50 > 1000 nM T82078 C4K8NM 56851182 EC50 > 1000 nM T82078 CLT65O 56851306 EC50 > 1000 nM T82078 CQH8R9 56851450 EC50 > 1000 nM T82078 C35ONK 57384785 EC50 = 1.01 nM T82078 C4ZY6M 57384786 EC50 = 1.64 nM T82078 CQ5Z0D 57384787 EC50 = 3.8 nM T82078 C1Z9CB 57384789 EC50 = 4.5 nM T82078 CU30HE 57388031 EC50 = 5.52 nM T82078 CB1VQ8 57388036 EC50 = 4.79 nM T82078 C4Y5XA 57740266 EC50 = 23 nM T82078 CH29GF 71258526 IC50 > 10000 nM T82078 CIB14T 71451937 Ki = 25 nM T82078 CPCT40 71451938 EC50 = 78 nM T82078 C83LQK 71453783 EC50 = 25 nM T82078 CZDG94 71457280 EC50 = 3.7 nM T82078 C2KRU3 71457309 EC50 = 56 nM T82078 CKQ03G 71462640 EC50 = 20 nM T82078 CGJ0Q1 118719088 Ki = 11 nM T82078 C45BQH 132585194 EC50 > 100000 nM T82078 CAVF95 137553173 EC50 = 0.11 nM T82078 CTP9M8 145968052 IC50 = 4651 nM T82078 COQ29Y 145968118 IC50 = 4363 nM T82078 C4T7FK 145968297 IC50 = 1682 nM T82078 CJ01EH 145968400 IC50 = 4755 nM T82078 CR8SB5 145968508 IC50 = 3373 nM T82078 CY6GD5 145969059 IC50 = 7519 nM T82078 CYQZ05 145969942 IC50 = 3938 nM T82078 CP50WV 145970164 IC50 = 1962 nM T82078 CE41IX 145987954 IC50 = 6427 nM T82078 CAKE87 149687120 EC50 = 1000 nM T82078 CRJ74Z 150370253 EC50 = 1350 nM T82078 CT2CO6 150457654 EC50 = 3000 nM T82078 C0GR6S 151417654 EC50 = 5000 nM T82078 CAC0J5 151485696 EC50 = 1450 nM T82078 CL7F2W 151543599 EC50 = 320 nM T82078 CAM64K 152550631 EC50 = 3090 nM T82078 CO94FB 152580191 EC50 = 45240 nM T82078 C1QR9N 152598982 EC50 = 6630 nM T82078 C67ORV 155514087 EC50 = 46.16 nM T82078 CN6IC3 155515837 EC50 = 0.304 nM T82078 C9L5GP 155519718 EC50 = 160 nM T82078 C3SNM6 155524646 EC50 = 150.6 nM T82078 CISL79 155528194 EC50 = 0.609 nM T82078 CAI06Z 155528951 EC50 = 3460 nM T82078 CUM0D7 155530294 EC50 = 161.01 nM T82078 CO8T1L 155533032 EC50 = 4590 nM T82078 C3YD6A 155534493 EC50 = 450 nM T82078 C7KV8W 155535367 EC50 = 11820 nM T82078 CL6A9D 155536490 EC50 = 16380 nM T82078 C74LZY 155537225 EC50 = 14160 nM T82078 C2NRE1 155548273 EC50 = 1.162 nM T82078 CW2V9Z 155548681 EC50 = 1330 nM T82078 CHSC79 155553471 EC50 = 0.383 nM T82078 C1Y6NK 155555507 EC50 = 0.281 nM T82078 CE1Q2L 155558171 EC50 = 0.468 nM T82078 CU7S9Z 155559013 EC50 = 155.69 nM T82078 CQ4I7V 155562153 EC50 = 4.445 nM T82078 C6H2TX 155562332 EC50 = 17.38 nM T82078 CSW73J 155564215 EC50 = 22.96 nM T82078 D02TVS 985 IC50 = 5000 nM T82078 D08OBF 11005 IC50 = 5000 nM T42319 CBC0J5 6418797 IC50 = 15 nM T42319 CC9S5U 28412206 IC50 = 160 nM T42319 C5MQR9 130365202 IC50 = 22 nM T03150 D0O1UZ 644019 IC50 > 100000 nM T03150 D0T9TJ 3034010 IC50 = 1 nM T03150 C3ERF2 30219 IC50 > 100000 nM T03150 CJ5T2N 98523 IC50 = 27300 nM T03150 C2DF6O 160570 IC50 = 19400 nM T03150 CZ46HG 5315659 IC50 > 100000 nM T03150 C2AR0Z 6449999 IC50 = 30500 nM T03150 CY6D5H 9821458 IC50 = 26.3 nM T03150 CNZ60S 9968521 IC50 = 25000 nM T03150 C48MPN 10445943 IC50 = 549.54 nM T03150 CU94ZT 11484453 IC50 > 10000 nM T03150 C4CN3F 11601669 IC50 = 16600 nM T03150 CG2B7X 11631387 IC50 > 10000 nM T03150 C57KVO 11674428 IC50 > 10000 nM T03150 CAG6H2 11709766 IC50 > 10000 nM T03150 CQ0U8Y 11991811 IC50 > 10000 nM T03150 C24DMZ 11991812 IC50 = 1819.7 nM T03150 CNS07O 11991890 IC50 > 10000 nM T03150 CE1C9H 11991893 IC50 > 10000 nM T03150 CAW97C 11991894 IC50 > 10000 nM T03150 CVK4C5 11991896 IC50 > 10000 nM T03150 CI9R2Y 11991988 IC50 > 10000 nM T03150 C89XWP 11991989 IC50 > 10000 nM T03150 C2GA4E 13817938 IC50 = 5000 nM T03150 CL93TQ 14847017 IC50 > 25000 nM T03150 CF1EO5 14852550 IC50 = 2800 nM T03150 CUO5V8 16110633 IC50 > 10000 nM T03150 C8HM0A 16110639 IC50 > 10000 nM T03150 CY41WJ 16110645 IC50 > 10000 nM T03150 CGY2J1 16110648 IC50 > 10000 nM T03150 C64TVY 16110650 IC50 > 10000 nM T03150 C9UE5X 16110705 IC50 > 10000 nM T03150 CS8QF4 16110720 IC50 > 10000 nM T03150 CKDP17 22486170 IC50 = 74.13 nM T03150 CG2UP9 22486172 IC50 = 64.57 nM T03150 C40ZRT 22486173 IC50 > 10000 nM T03150 C60VIC 22486175 IC50 = 74.13 nM T03150 C12FHJ 22486192 IC50 > 10000 nM T03150 C1IQ9L 22486206 IC50 = 46.77 nM T03150 CX38ZN 22848569 IC50 = 100 nM T03150 CC89OP 24795575 IC50 = 10000 nM T03150 CB20PL 24795576 IC50 = 510 nM T03150 C3FXH6 24795577 IC50 = 600 nM T03150 CA3F9Q 24795578 IC50 = 500 nM T03150 C0CR1M 24795717 IC50 = 4400 nM T03150 CZIU76 24795718 IC50 = 340 nM T03150 CUK3T7 24795721 IC50 = 200 nM T03150 CQ1V8D 24795722 IC50 = 570 nM T03150 C7OF2P 24795723 IC50 > 10000 nM T03150 CF1V5Z 24795854 IC50 > 10000 nM T03150 C0O2FX 24796127 IC50 = 10000 nM T03150 CWK84C 24796128 IC50 = 10000 nM T03150 C9FQD3 24796129 IC50 = 10000 nM T03150 CS0DM2 24798460 IC50 > 10000 nM T03150 CPB6D7 24948912 IC50 > 10000 nM T03150 C4R3EO 24948913 IC50 > 10000 nM T03150 C0MC4D 24948914 IC50 > 10000 nM T03150 CZ51NC 24948915 IC50 > 10000 nM T03150 CV0U8Z 24949074 IC50 > 10000 nM T03150 CGK9I3 24949076 IC50 > 10000 nM T03150 C2SZ3G 24949077 IC50 > 10000 nM T03150 CH0M1T 24949222 IC50 > 10000 nM T03150 CET9M4 24949223 IC50 = 2041.74 nM T03150 C8H3VQ 24949224 IC50 > 10000 nM T03150 C2SVE6 24949225 IC50 = 1047.13 nM T03150 CS8H1V 24950364 IC50 > 10000 nM T03150 CIY0F3 24950522 IC50 > 10000 nM T03150 C86RHX 24950524 IC50 > 10000 nM T03150 CO37IU 24950526 IC50 > 10000 nM T03150 CF63PK 24950527 IC50 > 10000 nM T03150 CU8Z1I 24950681 IC50 > 10000 nM T03150 CV3Q5X 24950682 IC50 > 10000 nM T03150 C42VIK 24950684 IC50 > 10000 nM T03150 C6TNZ0 24950685 IC50 > 10000 nM T03150 CLW02V 24951001 IC50 = 2754.23 nM T03150 CDEV57 24951002 IC50 = 933.25 nM T03150 CW1H7D 24951003 IC50 = 1949.84 nM T03150 C4MXB8 24951004 IC50 > 10000 nM T03150 CIF25O 24951005 IC50 > 10000 nM T03150 CFJW54 24951156 IC50 > 10000 nM T03150 C6O2UZ 24951157 IC50 > 10000 nM T03150 CA9XL1 24951158 IC50 > 10000 nM T03150 CSDT93 24951161 IC50 > 10000 nM T03150 C3GC9N 24951316 IC50 > 10000 nM T03150 CXH2N9 24951317 IC50 > 10000 nM T03150 CUDP87 24951320 IC50 > 10000 nM T03150 CD4P8C 24951321 IC50 > 10000 nM T03150 CW2T9Y 25140054 IC50 > 25000 nM T03150 CS0Z2Y 25140206 IC50 = 800 nM T03150 CX9OQ0 25140207 IC50 > 25000 nM T03150 C4U5PK 25140353 IC50 = 25000 nM T03150 CPB4N3 25140358 IC50 = 43 nM T03150 CDXE43 25140500 IC50 = 460 nM T03150 C3F4ZI 25140502 IC50 = 1100 nM T03150 CSY05H 25140504 IC50 > 25000 nM T03150 C01XPW 25140640 IC50 > 25000 nM T03150 C3J7SK 25140642 IC50 = 25000 nM T03150 CAH40Z 25224932 IC50 = 35 nM T03150 C3NRB0 44185423 IC50 > 25000 nM T03150 C8RTA7 44389776 IC50 = 3.631 nM T03150 CJ91NL 44391726 IC50 > 10000 nM T03150 C9KVQ5 44398776 IC50 = 2398.83 nM T03150 CRY47W 44448494 IC50 > 10000 nM T03150 CA49WS 44448505 IC50 > 10000 nM T03150 C6AY8U 44448506 IC50 > 10000 nM T03150 C7ZJ9O 44448536 IC50 > 10000 nM T03150 C72IYN 44448539 IC50 > 10000 nM T03150 CZTQ62 44448540 IC50 > 10000 nM T03150 C4G9YD 44448542 IC50 > 10000 nM T03150 CBA36L 44448576 IC50 > 10000 nM T03150 CSB9M8 44448577 IC50 > 10000 nM T03150 C0J4VA 44448578 IC50 > 10000 nM T03150 CGL3J5 44448579 IC50 > 10000 nM T03150 COWF13 44448613 IC50 > 10000 nM T03150 C7VGI3 44448615 IC50 > 10000 nM T03150 CIR53D 44448618 IC50 > 10000 nM T03150 CVB6E5 44448647 IC50 > 10000 nM T03150 CS9YA3 44448648 IC50 > 10000 nM T03150 C7JYR2 44448650 IC50 > 10000 nM T03150 CC1AM6 44452817 IC50 = 2238.72 nM T03150 C7D3IE 44554444 IC50 > 10000 nM T03150 CJ4BM8 44554447 IC50 = 123.03 nM T03150 C10PFH 44554611 IC50 > 10000 nM T03150 CL6C1X 44554613 IC50 > 10000 nM T03150 CUSY65 44554617 IC50 > 10000 nM T03150 CK87GF 44554786 IC50 = 3388.44 nM T03150 C6KCQ1 44554787 IC50 = 213.8 nM T03150 CSC92W 44563442 IC50 = 160 nM T03150 CP6T2X 44588588 IC50 = 600 nM T03150 CHI7K5 44588701 IC50 = 16 nM T03150 C21ZJU 44588702 IC50 = 430 nM T03150 CR15XH 44589030 IC50 > 25000 nM T03150 CE8S5M 44589338 IC50 = 204.17 nM T03150 CC3Y8W 45040160 IC50 = 0.2512 nM T03150 C8PJ6E 53354789 IC50 = 0.6 nM T03150 CYMP74 53354793 IC50 = 55 nM T03150 CFDZ53 53358485 IC50 = 3 nM T03150 CGA17H 53358723 IC50 = 3 nM T03150 CQP8H6 53364459 IC50 = 25.12 nM T03150 CG6O9T 53364485 IC50 = 125.89 nM T03150 C5U3CY 53364540 IC50 = 25.12 nM T03150 CTXO65 53371759 IC50 = 80 nM T03150 CKDV43 53371760 IC50 = 510 nM T03150 C63OKT 53371761 IC50 = 60 nM T03150 C2NPB3 53371884 IC50 = 4 nM T03150 C8A7NI 53371887 IC50 = 45 nM T03150 CT4JQ2 53371888 IC50 = 14000 nM T03150 C83XNU 53372007 IC50 = 161 nM T03150 CJF54L 53372010 IC50 = 8 nM T03150 CW4L5A 53372145 IC50 = 40 nM T03150 C3KG7Q 53372147 IC50 = 130 nM T03150 CXS23L 53373470 IC50 = 88 nM T03150 CT6K2O 53373472 IC50 = 82 nM T03150 C1LOV9 53373473 IC50 = 6 nM T03150 C3MZ8V 56593112 IC50 = 63.1 nM T03150 CS64LM 57519635 IC50 = 2.512 nM T03150 C3N9ZD 58408422 IC50 = 11 nM T03150 CI4BZ7 59444387 IC50 = 35000 nM T03150 C12DNA 59444416 IC50 > 50000 nM T03150 CVOT61 68856433 IC50 = 194.98 nM T03150 CUJ4Q7 97289144 IC50 = 39.81 nM T03150 CA0B1S 97289145 IC50 = 0.7943 nM T03150 C5DP6A 102340761 IC50 = 18 nM T03150 C3Q2YW 118709691 IC50 = 185 nM T03150 C1LD8T 118709692 IC50 = 56 nM T03150 CH68VA 118709693 IC50 = 143 nM T03150 C7WM1Y 118709694 IC50 = 65 nM T03150 CL7V1A 118709695 IC50 = 91 nM T03150 CEP4Y2 118709696 IC50 = 1600 nM T03150 CAJL96 118709697 IC50 = 66 nM T03150 C9LA4W 118709698 IC50 = 695 nM T03150 CO2UK4 118709699 IC50 > 10000 nM T03150 CJYP65 118709700 IC50 > 10000 nM T03150 COT9G8 118709701 IC50 = 302 nM T03150 C5OQW3 118709702 IC50 > 10000 nM T03150 CK3HD2 118709703 IC50 > 10000 nM T03150 CL8RB7 118709704 IC50 > 10000 nM T03150 C8QWB1 118709705 IC50 > 10000 nM T03150 CI9WT6 118709706 IC50 > 10000 nM T03150 C8A3LJ 118709707 IC50 > 10000 nM T03150 C13UNC 118709708 IC50 > 10000 nM T03150 CA2RM6 118709709 IC50 = 512 nM T03150 CWXU60 118709710 IC50 > 10000 nM T03150 C2CFK6 122390213 IC50 = 3.162 nM T03150 CUPL34 127025121 IC50 = 707.95 nM T03150 CVZ6L2 127025122 IC50 > 10000 nM T03150 COAV54 127025123 IC50 = 891.25 nM T03150 CE95CQ 127025124 IC50 = 5888.44 nM T03150 CLGM46 127025429 IC50 > 10000 nM T03150 CL59BD 127027280 IC50 > 10000 nM T03150 CD19CU 127028613 IC50 = 389.05 nM T03150 CD8A2G 127028614 IC50 = 478.63 nM T03150 CNM4G2 127034816 IC50 > 10000 nM T03150 CBNG31 127035005 IC50 = 87.1 nM T03150 C87QBE 127035301 IC50 > 10000 nM T03150 CRI8C3 127036608 IC50 > 10000 nM T03150 C3QY5D 127036781 IC50 = 18197.01 nM T03150 CO80TX 127036849 IC50 = 12022.64 nM T03150 C5AE4N 127036850 IC50 > 10000 nM T03150 C8QOD6 127036851 IC50 = 1230.27 nM T03150 CWH7V5 127036852 IC50 > 10000 nM T03150 C3J4PI 127036853 IC50 = 204.17 nM T03150 CJ8Q0R 127036854 IC50 = 1698.24 nM T03150 CP7JQ2 127036983 IC50 = 117.49 nM T03150 CDN8R0 127036984 IC50 = 1412.54 nM T03150 CNKM09 127037362 IC50 > 10000 nM T03150 CCT47B 127037865 IC50 = 30 nM T03150 CG6US2 127039578 IC50 = 18 nM T03150 CF6YI4 127039579 IC50 = 19 nM T03150 C48OAZ 127039864 IC50 = 0.9 nM T03150 CHT12Z 127039880 IC50 = 2.4 nM T03150 C83IWM 127039881 IC50 > 30000 nM T03150 CP5IT2 127039882 IC50 = 80 nM T03150 CPU6M7 127040547 IC50 = 13500 nM T03150 CT90IK 127040548 IC50 = 16000 nM T03150 CRY71W 127040549 IC50 = 3 nM T03150 C60HOC 127040550 IC50 = 17 nM T03150 CQB3W9 127041215 IC50 = 17 nM T03150 CMX21S 127041501 IC50 = 16 nM T03150 CEA48I 129188688 IC50 = 1.259 nM T03150 C49PJB 129188708 IC50 = 0.5012 nM T03150 CW1G0V 134131835 IC50 = 398.11 nM T03150 C2PYB4 134133861 IC50 = 7.943 nM T03150 CM4WT3 134133947 IC50 = 0.631 nM T03150 CS6VC7 134134749 IC50 = 19.95 nM T03150 C8NST5 134135610 IC50 = 5.012 nM T03150 CY32GJ 134136787 IC50 = 3981.07 nM T03150 CZW3T0 134138122 IC50 = 100 nM T03150 C2GX1J 134138767 IC50 = 12.59 nM T03150 CK7MS5 134139434 IC50 = 5.012 nM T03150 CTWL68 134140363 IC50 = 7.943 nM T03150 C3BWS0 134141954 IC50 = 12.59 nM T03150 CWES31 134142232 IC50 = 0.7943 nM T03150 CBA6M0 134142396 IC50 = 5.012 nM T03150 C4H7UW 134143500 IC50 = 19.95 nM T03150 CTZK53 134143949 IC50 = 0.7943 nM T03150 CYI16B 134145542 IC50 = 3.162 nM T03150 CCBN29 134147523 IC50 = 158.49 nM T03150 CU98PE 134149903 IC50 = 19.95 nM T03150 CMQ9L3 134150114 IC50 = 19.95 nM T03150 CU7D8C 134151520 IC50 = 5011.87 nM T03150 C2N3VI 134153875 IC50 = 1 nM T03150 CXYP40 134156008 IC50 = 1584.89 nM T03150 CSOX06 134156265 IC50 = 6.31 nM T03150 CKJ1X4 134157652 IC50 = 6309.57 nM T03150 CO1MF8 145979117 IC50 = 31.62 nM T03150 CBF8Z1 145979505 IC50 = 25.12 nM T03150 CPJ13H 145980248 IC50 > 10000 nM T03150 CZ5GX0 145980541 IC50 = 0.7943 nM T03150 C9ZVP4 145980767 IC50 = 79.43 nM T03150 C4CW1J 145981620 IC50 > 10000 nM T03150 CD5G1L 145982097 IC50 > 10000 nM T03150 C0T9PD 145982431 IC50 = 15.85 nM T03150 C9XUQ0 145983194 IC50 > 10000 nM T03150 C3IA4D 145986832 IC50 = 25.12 nM T03150 C8U1LO 145987585 IC50 = 79.43 nM T03150 CAH95K 145988033 IC50 > 10000 nM T03150 CSTI30 145988650 IC50 = 1258.93 nM T03150 CU1BT5 145989121 IC50 > 10000 nM T03150 CT0H4P 145990805 IC50 = 25.12 nM T03150 C1Z9EW 145990933 IC50 = 15.85 nM T03150 C3OXW0 145992126 IC50 > 10000 nM T03150 C3JMC7 145992455 IC50 > 10000 nM T03150 C4Q1ME 145992746 IC50 = 158.49 nM T03150 CXYG34 145993594 IC50 > 10000 nM T03150 CO67DP 145994122 IC50 = 15.85 nM T03150 CTA39R 155557726 IC50 = 690 nM T03150 D00CKY 24951315 IC50 > 10000 nM T03150 D01BGK 44554788 IC50 > 10000 nM T03150 D01JCJ 22486174 IC50 = 630.96 nM T03150 D02IQP 22486203 IC50 > 10000 nM T03150 D02JVI 44387731 IC50 = 3630.78 nM T03150 D03NTQ 24951319 IC50 > 10000 nM T03150 D03OGD 44554610 IC50 = 630.96 nM T03150 D03SCD 44448616 IC50 > 10000 nM T03150 D04JWW 44554441 IC50 = 2344.23 nM T03150 D05LXG 5063 IC50 = 60 nM T03150 D05MBJ 44554446 IC50 = 123.03 nM T03150 D06VSA 11991809 IC50 > 10000 nM T03150 D07GOA 11150976 IC50 = 524.81 nM T03150 D07QOG 44554445 IC50 = 1513.56 nM T03150 D0D7HU 24950683 IC50 > 10000 nM T03150 D0D8PZ 93147 IC50 > 50000 nM T03150 D0E0JC 11279040 IC50 > 10000 nM T03150 D0F9LO 44554440 IC50 = 2398.83 nM T03150 D0H5RS 11991808 IC50 > 10000 nM T03150 D0K6MH 25147546 IC50 = 575.44 nM T03150 D0K8MN 44448617 IC50 > 10000 nM T03150 D0KI3F 44554272 IC50 > 10000 nM T03150 D0PN9S 44554614 IC50 = 8709.64 nM T03150 D0Q2CR 24950841 IC50 = 2691.53 nM T03150 D0Q9JN 11991888 IC50 > 10000 nM T03150 D0TN0A 10085812 IC50 = 37.15 nM T03150 D0U3YC 44560315 IC50 = 130 nM T03150 D0U5LL 2543 IC50 > 50000 nM T03150 D0U8YV 24951000 IC50 > 10000 nM T03150 D0W7NY 11991895 IC50 > 10000 nM T03150 D0W7XR 11507802 IC50 > 10000 nM T03150 D0X6WV 44554442 IC50 > 10000 nM T03150 D0X8ZO 9972176 IC50 = 30.9 nM T47215 D06BEP 2712 IC50 = 100000 nM T47215 D07JVL 3016 IC50 > 100000 nM T47215 D0CP4E 2802 IC50 > 100000 nM T47215 D0W2NM 3380 IC50 > 100000 nM T47215 D02PSZ 9962628 IC50 = 3.7 nM T47215 D08AWI 11430856 Ki > 2000 nM T47215 CXI14V 196641 IC50 = 2400 nM T47215 C7SZ9E 613843 IC50 > 100000 nM T47215 C83EHQ 4259649 IC50 > 100000 nM T47215 CPM2W0 5279119 IC50 > 40000 nM T47215 CFR37P 5279123 IC50 > 40000 nM T47215 C3CT7R 5279366 IC50 = 23000 nM T47215 CESY43 5279395 IC50 > 100000 nM T47215 CF74HA 6918156 EC50 = 0.1 nM T47215 C65UQT 7216755 IC50 > 100000 nM T47215 CB80WJ 7216757 IC50 > 100000 nM T47215 CIT4S2 9865694 IC50 > 100000 nM T47215 C1IWA0 10001488 IC50 = 11000 nM T47215 CM81IO 10093957 IC50 = 300 nM T47215 CX97LH 10156187 IC50 > 40000 nM T47215 CFX06L 10182876 IC50 > 100000 nM T47215 CCFV43 10320031 IC50 = 11000 nM T47215 CA5B8O 10391834 EC50 = 210 nM T47215 C57AXJ 10440992 EC50 = 15 nM T47215 C1MTR3 10454890 IC50 = 3400 nM T47215 CT8H3X 10476766 IC50 = 3000 nM T47215 C91ZVY 10507109 EC50 = 1600 nM T47215 CQP20O 13809511 IC50 = 13000 nM T47215 CT20PV 13809514 IC50 > 40000 nM T47215 CCJ8B2 13972377 IC50 = 100000 nM T47215 CMF30H 14208192 IC50 = 8000 nM T47215 CZ05OR 14208194 IC50 = 3700 nM T47215 C9WM1D 14208197 IC50 > 100000 nM T47215 CNDY74 14208198 IC50 = 20000 nM T47215 CC28YX 14208199 IC50 = 8400 nM T47215 CS3GZ8 14208200 IC50 = 100000 nM T47215 C90NPA 14208201 IC50 > 100000 nM T47215 CEZ28U 14208202 IC50 = 3300 nM T47215 CNE6M7 14208204 IC50 = 40000 nM T47215 CCRZ68 14208205 IC50 = 80000 nM T47215 C95CUY 14208206 IC50 = 80000 nM T47215 CN26QE 14208208 IC50 = 5500 nM T47215 CUWX86 14208210 IC50 = 32000 nM T47215 CO0VN7 14208211 IC50 > 40000 nM T47215 CL68OI 14208212 IC50 > 40000 nM T47215 CYI95A 14208213 IC50 = 100000 nM T47215 COSQ82 14208214 IC50 = 12000 nM T47215 CD54MZ 14208215 IC50 = 12000 nM T47215 C4DFM9 14208216 IC50 = 26000 nM T47215 CX5QY0 14208217 IC50 > 50000 nM T47215 C31PLA 14208220 IC50 = 48000 nM T47215 C9PC8E 14208221 IC50 = 2700 nM T47215 C9HAS5 14208225 IC50 = 300 nM T47215 CD5EB1 14208226 IC50 = 1100 nM T47215 C1U8QJ 14208227 IC50 = 1000 nM T47215 CPON92 14208228 IC50 = 5600 nM T47215 C06SBR 14208229 IC50 = 12000 nM T47215 C61QZS 14208230 IC50 = 38000 nM T47215 CH7OP3 14208231 IC50 = 15000 nM T47215 C9M2XR 14208232 IC50 = 6000 nM T47215 CBU7Q1 14208233 IC50 = 50000 nM T47215 CY4SV8 14208234 IC50 = 16000 nM T47215 CJ9U4R 14208235 IC50 = 29000 nM T47215 CHZ4I8 14208236 IC50 = 7000 nM T47215 C2P6RF 14208237 IC50 = 200 nM T47215 CZV4C2 14208238 IC50 = 100000 nM T47215 CW3R9Q 14208239 IC50 = 100000 nM T47215 C6RHK0 14208240 IC50 > 50000 nM T47215 C8VAY7 14208241 IC50 = 2900 nM T47215 CZFH81 14208242 IC50 = 1900 nM T47215 C36GAC 14208243 IC50 = 40000 nM T47215 CX36ZB 14208245 IC50 > 40000 nM T47215 CY74SB 14208246 IC50 > 40000 nM T47215 C1UYA8 14208247 IC50 = 21000 nM T47215 CYO09N 14208248 IC50 = 40000 nM T47215 C8ZW3F 14208249 IC50 = 14000 nM T47215 C1ZE2W 14208250 IC50 > 100000 nM T47215 CGP9U0 14208251 IC50 = 22000 nM T47215 CDZ4I9 14208252 IC50 = 83000 nM T47215 C2IY4X 14208253 IC50 = 75000 nM T47215 CU8JZ3 14208254 IC50 > 40000 nM T47215 CRO59W 14208255 IC50 > 100000 nM T47215 CNH0M3 14208256 IC50 > 40000 nM T47215 CLMD93 14208257 IC50 > 40000 nM T47215 CA8ON0 14208258 IC50 = 43000 nM T47215 CXND36 14208259 IC50 = 3700 nM T47215 C9YEC6 14208260 IC50 = 65000 nM T47215 CDK6O7 14208261 IC50 = 12000 nM T47215 CT14KZ 14208262 IC50 = 18000 nM T47215 C1IDH6 14208263 IC50 = 8000 nM T47215 C84QFK 14208264 IC50 = 100000 nM T47215 C1J7OL 14208265 IC50 > 100000 nM T47215 C7U4EF 14208266 IC50 = 100000 nM T47215 CC6Q1J 14208267 IC50 > 100000 nM T47215 CEK7X0 14208268 IC50 = 2400 nM T47215 C3KC0H 14208269 IC50 = 1600 nM T47215 CD7M8S 14208270 IC50 = 2900 nM T47215 CU0R4P 14208271 IC50 = 1800 nM T47215 C81RHA 14208272 IC50 = 1400 nM T47215 C2AC0G 14208273 IC50 = 100000 nM T47215 CU8DT5 14208274 IC50 = 2300 nM T47215 C5Q4LT 14208275 IC50 = 8000 nM T47215 CQS07B 14208280 IC50 > 100000 nM T47215 C6V0OH 14208282 IC50 > 100000 nM T47215 CP2AD3 14208283 IC50 > 100000 nM T47215 C8IAW7 14208284 IC50 = 18000 nM T47215 C4AFQ0 14208286 IC50 = 640 nM T47215 CJ63WK 14208288 IC50 > 100000 nM T47215 C3IGO6 14208293 IC50 = 3500 nM T47215 CU5OL2 14208295 IC50 = 4000 nM T47215 CC1NM2 14208297 IC50 = 3000 nM T47215 CO4YF7 14208299 IC50 = 70000 nM T47215 CTIB05 14208300 IC50 = 5900 nM T47215 CGN9B4 14208302 IC50 = 31000 nM T47215 C7WR8Z 14208303 IC50 = 1700 nM T47215 CNI38M 14208305 IC50 = 2400 nM T47215 CNV32K 14208307 IC50 = 45000 nM T47215 CWDF64 14208308 IC50 = 3800 nM T47215 C61CHZ 14208309 IC50 > 100000 nM T47215 C8MK0S 14208310 IC50 > 100000 nM T47215 C9JB4Q 14208312 IC50 = 4600 nM T47215 C2X1WI 14208313 IC50 = 3300 nM T47215 COR29A 14208315 IC50 = 71000 nM T47215 CQDF03 14208317 IC50 = 16000 nM T47215 C9WQF0 14423345 IC50 > 100000 nM T47215 C91DYA 14539667 IC50 = 30 nM T47215 C3YXG7 14539668 IC50 = 100 nM T47215 C6V5XT 15167808 IC50 = 33000 nM T47215 C5FV4M 15167811 IC50 = 100000 nM T47215 CLN01M 15167812 IC50 = 18000 nM T47215 CGQ28U 15167816 IC50 = 3200 nM T47215 CI06RY 15637150 IC50 > 100000 nM T47215 CS4WQ9 15666988 EC50 = 0.99 nM T47215 C5I4LT 15667001 EC50 = 6.9 nM T47215 CDJF92 15667003 EC50 = 1.3 nM T47215 CXH92N 15667011 EC50 = 0.32 nM T47215 CHK6O5 15667012 EC50 = 3.7 nM T47215 C8FOJ2 15667013 EC50 = 3.7 nM T47215 CYA7D1 15667014 EC50 = 0.64 nM T47215 CHR57O 15667015 EC50 = 50 nM T47215 CY5QE8 15667016 EC50 = 0.7 nM T47215 C8P7RD 15667019 EC50 = 140 nM T47215 C52VKG 16144750 EC50 = 280 nM T47215 C0W6GO 16146266 EC50 = 150 nM T47215 C8O6FN 21120982 EC50 = 1.4 nM T47215 C4L3JO 44277972 IC50 = 2 nM T47215 C3AFJ8 44277974 IC50 = 600 nM T47215 CL0U7V 44277976 IC50 = 1000 nM T47215 CY5X6A 44277978 IC50 = 6000 nM T47215 CAYV07 44278203 IC50 = 200 nM T47215 C7JYT2 44278205 IC50 = 30 nM T47215 CAVP45 44278207 IC50 = 7000 nM T47215 CTG0R5 44278209 IC50 = 0.5 nM T47215 C8QTM3 44286377 IC50 = 5 nM T47215 CYV5Q9 44286378 IC50 = 128 nM T47215 CH6IU4 44286379 IC50 = 50 nM T47215 CF16UW 44286457 IC50 = 4.2 nM T47215 CBS5K8 44286707 IC50 = 10400 nM T47215 CGAL19 44286708 IC50 = 9 nM T47215 C80WRN 44287093 IC50 = 32 nM T47215 C3E8XF 44287095 IC50 = 35 nM T47215 C2NLY1 44287096 IC50 = 18 nM T47215 CS2EB1 44301168 IC50 = 81000 nM T47215 C25OPB 44301228 IC50 = 81000 nM T47215 CGIC64 44301269 IC50 = 54000 nM T47215 CHZE21 44301316 IC50 = 40000 nM T47215 CJLK17 44307266 EC50 = 28 nM T47215 CGE4Q1 44311593 IC50 = 100000 nM T47215 C05ZPL 44311626 IC50 > 100000 nM T47215 C5N7QT 44311642 IC50 = 35000 nM T47215 CBFJ81 44311923 IC50 = 2900 nM T47215 CCE47R 44311939 IC50 = 1000 nM T47215 C2K5WT 44311988 IC50 > 100000 nM T47215 CHP0A5 44312020 IC50 > 100000 nM T47215 CW5JD6 44312041 IC50 = 12000 nM T47215 C48FIX 44314735 IC50 = 1000 nM T47215 C65JVK 44314765 IC50 = 40 nM T47215 C9F2TU 44314836 IC50 = 10 nM T47215 CS72VK 44315012 IC50 = 100 nM T47215 COZ98N 44315045 IC50 = 2 nM T47215 CGW36X 44323354 IC50 = 100000 nM T47215 C92OSK 44323601 IC50 = 100000 nM T47215 COAF14 44327225 EC50 = 0.5 nM T47215 CPAX62 44327502 EC50 = 3.5 nM T47215 CXB5P4 44327506 EC50 = 4 nM T47215 C92SBQ 44327526 EC50 = 26 nM T47215 CZS19I 44327580 EC50 = 0.9 nM T47215 CYXH20 44327581 EC50 = 37 nM T47215 CORU67 44330731 EC50 = 71 nM T47215 CT7I5W 44330874 EC50 = 2.5 nM T47215 C4BI6P 44365263 EC50 = 5600 nM T47215 CHAZ51 44365304 EC50 = 300 nM T47215 CMV8Q7 44365359 EC50 = 110 nM T47215 CLS4N8 57390472 IC50 = 1500 nM T47215 CQ92LO 57393204 IC50 = 2100 nM T47215 C7VX8Q 73350067 EC50 = 104 nM T47215 CJL20E 136026556 IC50 = 49000 nM T47215 CH5Q9M 136026558 IC50 = 7000 nM T47215 CSZ21M 136026563 IC50 = 100000 nM T47215 C1K5YZ 136026564 IC50 = 100000 nM T47215 CCQ4D8 136026565 IC50 = 100000 nM T47215 D00SDJ 11237664 IC50 > 10000 nM T47215 D01FHK 3086453 IC50 = 0.3 nM T47215 D05QBF 443375 IC50 = 270 nM T47215 D05YZC 59751 IC50 = 800 nM T47215 D06DTT 193319 IC50 > 100000 nM T47215 D0I8AF 9833444 EC50 = 0.009 nM T47215 D0M6ZF 44278569 IC50 = 0.6 nM T73180 CY3TD6 3348132 Ki = 5 nM T73180 CMW3O0 71451330 Ki = 410 nM T73180 C9QS6E 71456659 Ki = 5 nM T73180 D01UNE 44580457 Ki = 0.23 nM T73180 D0B3UN 44580458 Ki = 18400 nM T73180 D0Y5IQ 44255320 IC50 = 5000 nM T09538 D05EJG 6305 IC50 > 5000 nM T09538 D0CF2Q 26879 IC50 > 5000 nM T09538 D0F8RA 2153 IC50 > 5000 nM T09538 D0R1CR 6140 IC50 > 5000 nM T09538 CVCE53 8465 IC50 > 100000 nM T09538 C30HVY 27944 Ki = 16000 nM T09538 C7H9AN 52780 IC50 > 100000 nM T09538 C4B9TI 69640 IC50 > 5000 nM T09538 CQ28ZE 317657 IC50 = 2160 nM T09538 CDCA05 586278 IC50 = 4800 nM T09538 C0NJ2B 645025 IC50 = 6510 nM T09538 CU1P5O 645853 IC50 = 1850 nM T09538 C0U7XK 646303 IC50 = 980 nM T09538 CRM9S6 674647 IC50 = 5710 nM T09538 CN06WE 685663 IC50 = 910 nM T09538 CA09QJ 715454 IC50 = 8600 nM T09538 CAVI24 776480 IC50 = 1300 nM T09538 COJ04E 839345 IC50 = 43 nM T09538 C7IW4S 850030 IC50 = 1130 nM T09538 C83WMP 893397 IC50 = 1060 nM T09538 C5UAR2 910374 IC50 = 4580 nM T09538 CNR2B4 934901 IC50 = 1130 nM T09538 C8SZX0 940183 IC50 = 44 nM T09538 C83UKT 1223927 IC50 = 42000 nM T09538 CVK03C 1515366 IC50 = 8000 nM T09538 C69SXL 2931238 IC50 = 230 nM T09538 C9B3AM 2940433 IC50 = 29200 nM T09538 CAX45S 3332652 IC50 = 6140 nM T09538 C6R9GN 3668507 IC50 = 84 nM T09538 CW7YG3 3724041 IC50 = 8240 nM T09538 C4HGA6 4679684 IC50 = 6 nM T09538 CNH58V 6471866 IC50 = 1490 nM T09538 CVXA89 6472157 IC50 = 500 nM T09538 CP8LS2 6472404 IC50 = 1550 nM T09538 CA80ZY 6472631 IC50 = 690 nM T09538 CNUM85 6472703 IC50 = 1680 nM T09538 C91AHZ 6473097 IC50 = 510 nM T09538 CRQW69 7938148 IC50 = 6590 nM T09538 CWQ8T0 7938664 IC50 > 10000 nM T09538 CXS5U7 9267841 IC50 = 540 nM T09538 C9KGH4 13224102 IC50 = 3580 nM T09538 C08PXE 16418617 IC50 > 200000 nM T09538 CYG35L 16418622 IC50 = 3570 nM T09538 C7KO2S 16654595 IC50 = 1290 nM T09538 C9C4MT 16654607 IC50 = 500 nM T09538 CNQ1X4 16654644 IC50 = 120 nM T09538 CGK96T 16654645 IC50 > 10000 nM T09538 C01JOY 16654701 IC50 > 10000 nM T09538 CK86ZI 16654723 IC50 > 10000 nM T09538 CVZI93 16654877 IC50 = 10300 nM T09538 CQ3G1X 16749996 IC50 > 100000 nM T09538 CU31QP 16760951 IC50 = 7360 nM T09538 CJOC50 17590947 IC50 = 2590 nM T09538 CA5F1C 19509988 IC50 = 44 nM T09538 CIR47C 19509990 IC50 = 82 nM T09538 CS96IU 19510029 IC50 = 51 nM T09538 C3XQF8 19510137 IC50 = 46 nM T09538 CEWS46 20230376 IC50 = 10300 nM T09538 CG19LI 23342610 IC50 = 1510 nM T09538 CQK26M 24178126 IC50 = 119 nM T09538 C2X1NY 24178130 IC50 = 324 nM T09538 CFI8Q2 24178131 IC50 = 4850 nM T09538 C40RUL 24178133 IC50 = 574 nM T09538 CJ2CX1 24178134 IC50 = 828 nM T09538 CNX7Q5 24178135 IC50 = 488 nM T09538 C5U6BE 24178136 IC50 = 375 nM T09538 C57TOU 24178138 IC50 = 398 nM T09538 CVG4X3 24178139 IC50 = 1450 nM T09538 CCG8A3 24178141 IC50 = 100 nM T09538 C0BKF2 24178164 IC50 > 10000 nM T09538 CFCN59 24178168 IC50 = 134 nM T09538 CP0C9G 24178169 IC50 = 35 nM T09538 CKQ84Y 24178170 IC50 = 5 nM T09538 CECB26 24178176 IC50 = 459 nM T09538 C6R2NG 24178177 IC50 = 47 nM T09538 C52CPA 24178178 IC50 = 31 nM T09538 CAB97E 24178179 IC50 = 35 nM T09538 C8T6FV 24178180 IC50 = 285 nM T09538 CS5JK8 24178183 IC50 = 127 nM T09538 CIM0D7 24178184 IC50 = 56 nM T09538 C5S1NR 24178187 IC50 > 10000 nM T09538 CQ1BH7 24178213 IC50 = 650 nM T09538 COJ25L 24790972 IC50 > 100000 nM T09538 C94GLB 24790973 IC50 > 100000 nM T09538 C0AO2Q 24790974 IC50 > 100000 nM T09538 C3G1XL 24790980 IC50 > 100000 nM T09538 CN98AX 24790981 IC50 > 100000 nM T09538 C2TI0S 24790992 IC50 > 100000 nM T09538 CY51VS 24792834 IC50 > 100000 nM T09538 C8UX3E 25067478 IC50 = 8700 nM T09538 C95BPI 25067480 IC50 = 47500 nM T09538 C40DVS 25067482 IC50 > 100000 nM T09538 C7RI9A 25067484 IC50 > 100000 nM T09538 CM1SX9 25067486 IC50 = 93800 nM T09538 C8FBY2 25067488 IC50 > 100000 nM T09538 CJY6Z4 25067490 IC50 > 100000 nM T09538 CDJX98 25067492 IC50 = 78300 nM T09538 CG3LC6 25067494 IC50 = 18000 nM T09538 CN67WC 25067496 IC50 = 26300 nM T09538 C0AIS7 25067498 IC50 = 41100 nM T09538 C4VM7G 25199538 IC50 > 100000 nM T09538 CFB7T2 44541246 IC50 = 740 nM T09538 CJ0SN5 44541247 IC50 = 3160 nM T09538 C0S3UO 46341316 IC50 > 100000 nM T09538 CA51TP 46341321 IC50 > 100000 nM T09538 CY1L4W 47001115 IC50 = 3550 nM T09538 C0EFT7 50876360 IC50 = 4170 nM T09538 C53USQ 50919364 IC50 > 100000 nM T09538 CQ0B3Y 50919367 IC50 = 35000 nM T09538 CGP5Y7 50919368 IC50 > 100000 nM T09538 CAHS24 50919371 IC50 > 100000 nM T09538 CJ4U0P 50919372 IC50 = 81000 nM T09538 C6PZS1 50919375 IC50 > 100000 nM T09538 C0WH9T 50919378 IC50 = 74000 nM T09538 C56ESL 50919379 IC50 > 100000 nM T09538 C75AFE 51035363 IC50 > 100000 nM T09538 CO2GR6 51035365 IC50 = 37000 nM T09538 C3RNJ6 51035366 IC50 > 100000 nM T09538 CLUO75 51035367 IC50 > 100000 nM T09538 CFQW32 53245527 IC50 > 100000 nM T09538 CA7W0D 53245529 IC50 > 100000 nM T09538 CJ7AH8 53245532 IC50 > 100000 nM T09538 CGI97B 53245533 IC50 > 100000 nM T09538 CV3N6A 53245539 IC50 > 100000 nM T09538 CK4MW7 53245545 IC50 > 100000 nM T09538 C9M2VB 53245562 IC50 > 100000 nM T09538 CLF78S 53245566 IC50 > 100000 nM T09538 CS8HB0 53245567 IC50 = 96000 nM T09538 C95LAC 53245601 IC50 > 100000 nM T09538 C4XE0F 53245605 IC50 > 100000 nM T09538 C1KYP7 53245607 IC50 > 100000 nM T09538 CS4VA9 53301944 IC50 > 100000 nM T09538 CEF7A6 53301950 IC50 > 100000 nM T09538 C10SFI 53301952 IC50 > 100000 nM T09538 C2TVZ8 53301954 IC50 > 100000 nM T09538 CA1L0I 53301967 IC50 > 100000 nM T09538 CY1RD8 53301975 IC50 > 100000 nM T09538 C9Y7FB 53384787 IC50 > 100000 nM T09538 CY7U5Z 56684170 IC50 = 322 nM T09538 CQS31W 56684192 IC50 = 432 nM T09538 CM9O7C 56684219 IC50 = 671 nM T09538 CI9F0D 56684226 IC50 = 198 nM T09538 CXH0Q3 56684231 IC50 = 876 nM T09538 CC1L0U 56684238 IC50 = 1490 nM T09538 C1RF5W 56684239 IC50 = 147 nM T09538 C3Z7VT 56684281 IC50 = 1510 nM T09538 C14YGH 56684290 IC50 = 160 nM T09538 CXV9G0 76310601 IC50 > 100000 nM T09538 CO0RD4 76310602 IC50 > 100000 nM T09538 C0VGL8 76314235 IC50 > 100000 nM T09538 CK4P0M 76314236 IC50 > 100000 nM T09538 C3TNU8 76317808 IC50 > 100000 nM T09538 CX4T6P 76317809 IC50 > 100000 nM T09538 CI5S6R 76317810 IC50 > 100000 nM T09538 C24EIR 76325122 IC50 > 100000 nM T09538 CY47FJ 76328685 IC50 > 100000 nM T09538 C13DAF 76328686 IC50 > 100000 nM T09538 C06IQM 76328687 IC50 > 100000 nM T09538 C9AC4S 76328688 IC50 > 100000 nM T09538 CRW30Y 76332363 IC50 > 100000 nM T09538 C46HOG 76335991 IC50 > 100000 nM T09538 CLO5E6 89768280 IC50 = 73 nM T09538 C9NEA7 89768286 IC50 = 16 nM T09538 CX3DI6 89768289 IC50 = 65 nM T09538 CT8YV9 89768307 IC50 = 73 nM T09538 C5JPX9 89768344 IC50 = 310 nM T09538 CN4M0V 89768386 IC50 = 26 nM T09538 C9YKL5 89768408 IC50 = 19 nM T09538 C8VW3O 89768435 IC50 = 14 nM T09538 C8GS4O 89768436 IC50 = 109 nM T09538 C6FOJ5 89768486 IC50 = 193 nM T09538 C08SUF 89768573 IC50 = 16000 nM T09538 C3U9CI 89768585 IC50 = 178 nM T09538 CQO0B2 89768682 IC50 = 38 nM T09538 CBH64G 89775256 IC50 = 120 nM T09538 C2G8RW 89775258 IC50 = 1560 nM T09538 C7P3LU 89775325 IC50 = 183 nM T09538 CIV27X 89775349 IC50 = 73 nM T09538 CU8GR6 98201958 IC50 = 660 nM T09538 C7HM4S 98201960 IC50 = 4040 nM T09538 CM1QX6 132584225 IC50 = 13300 nM T09538 C9BD8V 137632708 IC50 = 1420 nM T09538 CSL68C 137632786 IC50 = 9370 nM T09538 C7H5WC 137634253 IC50 = 1330 nM T09538 CP85TI 137636579 IC50 = 850 nM T09538 CTQW80 137639392 IC50 = 2520 nM T09538 CDNM08 137640888 IC50 = 17600 nM T09538 C0Y4BN 137641016 IC50 = 2510 nM T09538 CM9J2H 137641189 IC50 = 2590 nM T09538 CQ6V8J 137642208 IC50 = 7710 nM T09538 C2UHR1 137642382 IC50 = 2420 nM T09538 CM0VW9 137642465 IC50 = 1330 nM T09538 CB9LO1 137643174 IC50 = 3530 nM T09538 C2BJ0P 137644233 IC50 = 920 nM T09538 C89UKS 137645647 IC50 = 1640 nM T09538 CB71FA 137646257 IC50 = 9230 nM T09538 C1W0BC 137647100 IC50 = 2470 nM T09538 CSO31A 137649365 IC50 = 2540 nM T09538 CJ2X9P 137649542 IC50 = 1170 nM T09538 CO7QK2 137649680 IC50 = 1940 nM T09538 C4J7OX 137649851 IC50 = 1070 nM T09538 CVK64S 137651950 IC50 = 1250 nM T09538 CP7I1D 137653596 IC50 = 920 nM T09538 C79CVJ 137653769 IC50 = 3690 nM T09538 CB8WM7 137654951 IC50 = 2310 nM T09538 CL3D5W 137656119 IC50 = 1830 nM T09538 CQ9IW4 137657455 IC50 = 580 nM T09538 C6S9LY 137658048 IC50 = 8370 nM T09538 CWT81N 137658105 IC50 = 9010 nM T09538 CGH5C8 137659171 IC50 = 2560 nM T09538 C9LP5I 137660262 IC50 = 6380 nM T09538 CHW39D 137660646 IC50 = 1990 nM T09538 CIX9B8 145977005 IC50 = 134 nM T09538 CWKM51 145979441 IC50 = 17700 nM T09538 CA0J2N 145979703 IC50 = 540 nM T09538 C50ZPR 145979899 IC50 = 2360 nM T09538 CC5D8M 145980184 IC50 = 290 nM T09538 CL75VW 145980413 IC50 = 880 nM T09538 CM1R6F 145980749 IC50 = 3190 nM T09538 C4WC9R 145981028 IC50 = 2020 nM T09538 C1UL9Q 145981323 IC50 = 250 nM T09538 C69YPI 145981525 IC50 = 1390 nM T09538 CU10RQ 145981673 IC50 = 620 nM T09538 CDQ0T6 145981705 IC50 = 5430 nM T09538 CKNS82 145982359 IC50 > 200000 nM T09538 CO0KC4 145983428 IC50 = 1430 nM T09538 CXA9K5 145984158 IC50 = 1530 nM T09538 C8WE1U 145984874 IC50 = 610 nM T09538 CNZ81D 145984900 IC50 = 3480 nM T09538 C3QF8N 145986829 IC50 > 100000 nM T09538 CE8N3X 145987231 IC50 = 1070 nM T09538 CF79AH 145987426 IC50 = 930 nM T09538 C3PGA7 145987876 IC50 = 1440 nM T09538 C3F7ZP 145988073 IC50 = 1060 nM T09538 CLH8M7 145988443 IC50 = 330 nM T09538 C87AJL 145988932 IC50 = 11120 nM T09538 C26SUT 145989162 IC50 = 280 nM T09538 CG43SV 145989741 IC50 > 100000 nM T09538 C9HR2G 145989930 IC50 > 200000 nM T09538 C9ORM6 145990052 IC50 = 1980 nM T09538 C0J5HR 145990471 IC50 > 200000 nM T09538 CVWI49 145990949 IC50 = 19100 nM T09538 C34IHB 145991003 IC50 = 210 nM T09538 C9N0WB 145991049 IC50 = 4520 nM T09538 C4YD8B 145991232 IC50 = 1120 nM T09538 CTQ21M 145991361 IC50 = 7860 nM T09538 CPT2X4 145991492 IC50 = 450 nM T09538 CVM93K 145991559 IC50 > 100000 nM T09538 CE03ZX 145991579 IC50 > 200000 nM T09538 CGV5K1 145991886 IC50 = 1530 nM T09538 CVO92P 145992144 IC50 = 380 nM T09538 CPI0F4 145992202 IC50 = 26400 nM T09538 C6PI7B 145992264 IC50 = 1350 nM T09538 CFW27N 145992560 IC50 = 4910 nM T09538 CD2VR0 145992920 IC50 = 560 nM T09538 CI4C2R 145992946 IC50 = 5780 nM T09538 CJ39WG 145993183 IC50 = 1150 nM T09538 CR7A8S 145993335 IC50 = 520 nM T09538 CD8IY4 145993630 IC50 = 1580 nM T09538 CCE09D 145993780 IC50 = 520 nM T09538 C4QID1 145993905 IC50 = 2590 nM T09538 D0F8VS 9085 IC50 > 5000 nM T09538 D0W4MZ 6106 IC50 > 5000 nM T74977 D0Y9ZE 4197 Ki > 100000 nM T74977 D02UFQ 11620908 IC50 > 10000 nM T74977 D03HUX 49792852 IC50 > 10000 nM T74977 D0HY9S 73386890 Ki = 0.11 nM T74977 D0J6RV 71599640 IC50 = 0.34 nM T74977 D0O0LS 25141092 IC50 > 10000 nM T74977 D0PO8N 117881270 IC50 = 5 nM T74977 CO2Y3R 3698 Ki = 80800 nM T74977 CK8R2P 119131 Ki = 98100 nM T74977 C61YBI 300385 IC50 = 12000 nM T74977 CQ01JA 322353 Ki > 1000000 nM T74977 C9LA1E 11486283 IC50 > 10000 nM T74977 CI8CR3 11623444 Ki = 5400 nM T74977 CZ25EP 11631251 Ki > 100000 nM T74977 C6LK9N 11646783 Ki = 4800 nM T74977 C86IBL 12799331 Ki > 100000 nM T74977 CP4C7R 12799333 Ki > 100000 nM T74977 C0QGS1 13942472 Ki = 91200 nM T74977 C5VPH9 16129448 IC50 = 991 nM T74977 C5M1EL 20399253 Ki = 25600 nM T74977 C3XI0R 23339828 Ki = 236400 nM T74977 CQEV29 24992861 IC50 = 241 nM T74977 CCM43R 25181368 Ki = 128200 nM T74977 CG1XA0 25195352 IC50 = 1746 nM T74977 CEL61X 44229839 IC50 > 10000 nM T74977 C6G2EC 44232693 IC50 > 11000 nM T74977 C13QXB 44236351 IC50 = 500 nM T74977 CJ37DI 44236353 IC50 = 2170 nM T74977 C97CDF 44555517 IC50 = 19 nM T74977 CY2GA6 44555518 IC50 = 72 nM T74977 CPV8A6 44555519 IC50 = 103 nM T74977 C9Q8VR 44555761 IC50 = 525 nM T74977 C68LVU 44555820 IC50 = 21 nM T74977 CP6FY8 44556163 IC50 = 84 nM T74977 CHA25B 44556214 IC50 = 36 nM T74977 CR2CH3 44556329 IC50 = 33 nM T74977 CMU45C 46886960 IC50 = 66 nM T74977 C5G2VE 46909588 IC50 = 1.8 nM T74977 CM9KV3 46927221 IC50 = 1 nM T74977 CUBE41 46927300 IC50 = 3 nM T74977 CYP7I9 46927301 IC50 = 1 nM T74977 C85UXG 46927371 IC50 = 14 nM T74977 CJKG69 46927447 IC50 = 360 nM T74977 CF91RS 49843531 IC50 > 10000 nM T74977 CE9QJ4 50914591 IC50 = 35 nM T74977 CC0AT3 50914874 IC50 = 39 nM T74977 C1VML8 52936434 Ki = 2900 nM T74977 CRL93S 52947958 IC50 = 1218 nM T74977 CZ3QU8 53234663 IC50 = 1 nM T74977 C1CR6S 53363307 IC50 = 823 nM T74977 CK03PA 53363389 IC50 = 146 nM T74977 CX7B5T 53389592 IC50 = 2600 nM T74977 C3DR5F 53476530 IC50 = 4300 nM T74977 CTH0B1 53476531 IC50 = 600 nM T74977 CF2LI9 53476532 IC50 = 640 nM T74977 C7M1JN 53476533 IC50 = 280 nM T74977 CFRA47 54675539 IC50 = 10 nM T74977 CG4WB5 54675542 IC50 = 7.93 nM T74977 C1QYV4 54675574 IC50 = 3.06 nM T74977 CXIZ08 56659726 IC50 = 391 nM T74977 CB3Q1P 56663194 IC50 = 206 nM T74977 CZYH57 56666592 IC50 = 530 nM T74977 C2BL7S 56676833 IC50 > 12000 nM T74977 CS3EP0 56676834 IC50 = 140 nM T74977 CRG16Y 56676835 IC50 = 130 nM T74977 C6B1PU 56676891 IC50 = 202 nM T74977 CIV57W 56947168 IC50 = 4810 nM T74977 CR16SD 56947170 IC50 = 8470 nM T74977 CP8J4Y 56973724 IC50 = 35 nM T74977 CPJX47 57111159 Ki = 30200 nM T74977 CX5L3P 57379119 IC50 = 130 nM T74977 CF0G7A 57381882 IC50 = 1 nM T74977 C7C8IS 57382314 IC50 = 58 nM T74977 CACW05 57386803 IC50 = 3060 nM T74977 CG14VM 57387301 IC50 = 7120 nM T74977 C2W0OD 58539094 Ki = 25 nM T74977 CQTB49 58692572 Ki > 100000 nM T74977 C5VY6S 66546721 IC50 = 260 nM T74977 CMT23K 66546905 IC50 = 28 nM T74977 C2HO8D 66547424 IC50 = 4 nM T74977 CJ5HI6 66547425 IC50 = 3 nM T74977 CLWU09 66547597 IC50 = 20 nM T74977 C6SFP7 66547759 IC50 = 860 nM T74977 CM4PW9 66548104 IC50 = 22 nM T74977 C8ZJF7 66548458 IC50 = 26 nM T74977 CZ0KN3 66548460 IC50 = 92 nM T74977 CGW4L5 66548650 IC50 = 79 nM T74977 C7Q2CM 66548653 IC50 = 460 nM T74977 CI41NJ 66548849 IC50 = 16 nM T74977 CTJ64B 66548850 IC50 = 58 nM T74977 CL75SB 66598559 IC50 = 4.2 nM T74977 CA90HX 66598613 IC50 = 7.5 nM T74977 CWK2M7 66598658 IC50 = 6.2 nM T74977 C7UX1A 66603863 IC50 = 0.7 nM T74977 C2VW9Z 66695602 IC50 = 2.8 nM T74977 C20UYG 66734432 IC50 = 5000 nM T74977 CK80LJ 67130050 IC50 = 2160 nM T74977 CU2OT4 67453293 IC50 = 390 nM T74977 C3A6XO 67453604 IC50 = 250 nM T74977 CM0J9N 67453714 IC50 = 17 nM T74977 C9YDU0 67453874 IC50 = 25 nM T74977 CJ17AL 67454461 IC50 = 2600 nM T74977 CQ07OH 67454621 IC50 = 380 nM T74977 C0TGF6 67454968 IC50 = 18 nM T74977 C27GKJ 67455273 IC50 = 16 nM T74977 CAS7C4 67455813 IC50 = 39 nM T74977 C6VUN5 67456033 IC50 = 340 nM T74977 C16UFQ 67456579 IC50 = 310 nM T74977 C3E2VF 67457022 IC50 = 90 nM T74977 C1DJ2X 67457636 IC50 = 80 nM T74977 C58CPG 67462136 IC50 = 550 nM T74977 C9GIH3 67465029 IC50 = 16 nM T74977 CZ4EY3 67974488 IC50 = 1.4 nM T74977 CS7H9Y 68229500 IC50 = 4 nM T74977 C8L4UO 68229585 IC50 = 33 nM T74977 C4M9YZ 68229762 IC50 = 980 nM T74977 C4BQ5O 68229839 IC50 = 340 nM T74977 CC29SY 68230037 IC50 = 580 nM T74977 C9D3SQ 68230705 IC50 = 90 nM T74977 C32TVX 68230798 IC50 = 3.5 nM T74977 CUR2V0 68290592 IC50 = 23 nM T74977 C7U4VX 68290829 IC50 = 63 nM T74977 C24IRX 68290838 IC50 = 15 nM T74977 C2SLT0 68290849 IC50 = 51 nM T74977 CY60FW 68290875 IC50 = 13 nM T74977 C7GK8I 68290918 IC50 = 8 nM T74977 CC8IR2 68290919 IC50 = 120 nM T74977 CVB70Q 68291007 IC50 = 21 nM T74977 CN3YX2 68291016 IC50 = 7 nM T74977 C0OIP9 68291028 IC50 = 20 nM T74977 C7CZX6 68291099 IC50 = 27 nM T74977 CEJ26R 68291131 IC50 = 25 nM T74977 CEZI21 68291184 IC50 = 20 nM T74977 CY5OU4 68291366 IC50 = 71 nM T74977 C8CSV6 68291375 IC50 = 25 nM T74977 C2S0CH 68291448 IC50 = 74 nM T74977 C2ZLY3 68310278 IC50 = 600 nM T74977 CY4GV3 68310582 IC50 = 11 nM T74977 CLK8J5 68452965 IC50 = 1 nM T74977 CGE03L 68456113 IC50 = 4 nM T74977 CBE5C8 68525981 IC50 = 9 nM T74977 CR4XY0 68749727 IC50 = 9 nM T74977 C1KXF6 68750986 IC50 = 3 nM T74977 CSD73O 68750996 IC50 = 5 nM T74977 CTY35O 68753572 IC50 = 4 nM T74977 C7GRV2 68755406 IC50 = 1840 nM T74977 CTB87U 68756546 IC50 = 11 nM T74977 CER1B9 69093374 Ki = 150 nM T74977 CGTU20 69180001 IC50 = 35 nM T74977 CKX9D0 69180122 IC50 = 2 nM T74977 CC6W9E 69180323 IC50 = 7 nM T74977 C9IG3Y 69180487 IC50 = 28 nM T74977 C4SL6P 69181135 IC50 = 2 nM T74977 C19QYF 69181497 IC50 = 3 nM T74977 C4SKN0 69181574 IC50 = 1 nM T74977 CFHB37 70681991 IC50 = 1000 nM T74977 CCR5K4 70681992 IC50 = 5 nM T74977 CWK7B0 70682875 IC50 = 11 nM T74977 CY4JE7 70684107 IC50 = 130 nM T74977 C2Z6JE 70684108 IC50 = 3 nM T74977 CE1S5B 70686248 IC50 = 170 nM T74977 C68RKI 70686252 IC50 = 4 nM T74977 CI0FN3 70688373 IC50 = 5 nM T74977 C97YDW 70688374 IC50 = 7 nM T74977 CBYN07 70688375 IC50 = 4 nM T74977 CT47RZ 70690388 IC50 = 230 nM T74977 C39PBG 70692558 IC50 = 3 nM T74977 CC0W2L 70694608 IC50 = 510 nM T74977 CW75OG 70696648 IC50 = 9 nM T74977 CNA9E0 70696649 IC50 = 4 nM T74977 CEBO91 71452977 IC50 > 10000 nM T74977 C2XZO0 71576779 IC50 = 3.67 nM T74977 CZ31PU 71583657 IC50 > 10000 nM T74977 CHX9O7 71681990 IC50 = 438 nM T74977 CLK30W 71681991 IC50 = 116 nM T74977 C2EYU1 71682140 IC50 = 189 nM T74977 C9LG1S 71682141 IC50 = 28 nM T74977 CR3HA9 71682142 IC50 = 17 nM T74977 CU8BD4 71682143 IC50 = 32 nM T74977 C5OM4V 71682298 IC50 = 173 nM T74977 CH2RN0 71682299 IC50 = 2070 nM T74977 CP56ZV 71682300 IC50 = 119 nM T74977 CJ4B7I 71682457 IC50 = 12 nM T74977 CH9I6O 71735119 IC50 = 0.7 nM T74977 C7DFW5 71735277 IC50 = 0.4 nM T74977 C9SIU7 71735440 IC50 = 0.6 nM T74977 CEF5J3 71735441 IC50 = 0.7 nM T74977 CC6SF1 71737500 IC50 = 0.3 nM T74977 CD4W1T 72724724 IC50 = 28 nM T74977 CU15LG 72724725 IC50 > 100 nM T74977 C6OQ8P 72724726 IC50 = 46 nM T74977 CW87JM 72724727 IC50 = 22 nM T74977 C0J5IX 72724728 IC50 = 20 nM T74977 C10NMG 72724729 IC50 > 100 nM T74977 CAYC60 72724793 IC50 = 32 nM T74977 C47EPR 72724794 IC50 > 100 nM T74977 CY2K1G 72724795 IC50 > 100 nM T74977 C6U1XD 72724796 IC50 > 100 nM T74977 COC90M 72724797 IC50 = 12 nM T74977 CX3PH0 72724798 IC50 = 9 nM T74977 CD3Y8W 72724868 IC50 = 5 nM T74977 C1MXI3 72724869 IC50 = 8 nM T74977 CT64QU 72724870 IC50 = 2 nM T74977 CG12UO 72725640 IC50 > 100 nM T74977 C8QLX0 72725641 IC50 = 35 nM T74977 CZ8H4G 73345836 IC50 = 498 nM T74977 CUN62S 73386761 IC50 = 3660 nM T74977 CYFU24 73386762 IC50 = 660 nM T74977 C78QCA 73386764 IC50 = 99 nM T74977 C8MFJ1 73386768 IC50 = 8 nM T74977 CKW6Z2 73386776 IC50 = 150 nM T74977 CCS3G1 73386781 Ki = 24 nM T74977 C7ZRY0 73386874 IC50 = 18 nM T74977 CPZT25 73386878 Ki = 1.3 nM T74977 C9T0EL 73386880 Ki = 2.8 nM T74977 C01QMB 73386881 Ki = 4.2 nM T74977 CE2Y0X 73386882 Ki = 0.2 nM T74977 C4X5SL 73386970 IC50 = 110 nM T74977 C40ESH 73386976 IC50 = 24 nM T74977 CT18QV 73387064 Ki = 0.44 nM T74977 C5Y1IQ 73387066 IC50 = 46 nM T74977 CY52PU 73387073 Ki <= 0.07 nM T74977 CX6B4V 73387151 Ki = 0.094 nM T74977 CI1UR9 73387152 Ki = 0.13 nM T74977 CLZ7Q2 73670208 IC50 = 1.2 nM T74977 C47JPV 75202872 Ki = 0.77 nM T74977 C83YCN 75202873 IC50 = 5.8 nM T74977 CZS5U3 75203379 IC50 = 8.4 nM T74977 C76NUH 76310311 IC50 = 17 nM T74977 CP8F0T 76313983 IC50 = 160 nM T74977 C81ECP 76313984 IC50 = 28 nM T74977 C7HYN3 76313985 IC50 = 1600 nM T74977 CRLG27 76317532 IC50 = 4400 nM T74977 CH8Q9D 76324874 IC50 = 640 nM T74977 CN15WO 76328435 IC50 = 4900 nM T74977 C58NAD 76335737 IC50 = 32 nM T74977 C3HBX9 76335738 IC50 = 21 nM T74977 CS0CN8 76335739 IC50 = 990 nM T74977 C0RXT8 78320750 IC50 = 0.63 nM T74977 C9G0DM 86651966 IC50 = 12000 nM T74977 COW7F1 86711021 IC50 = 16 nM T74977 C53FOY 86711045 IC50 = 9.4 nM T74977 C3SQ6G 87057562 IC50 = 5.6 nM T74977 C8OSN4 89509786 IC50 = 4.1 nM T74977 C7CQD4 89971933 IC50 = 2.8 nM T74977 C2AM6R 89995977 IC50 = 250 nM T74977 CQL6V2 89995979 IC50 = 140 nM T74977 CB1M6J 89995980 IC50 = 10 nM T74977 CJ67CI 89995984 IC50 = 49 nM T74977 C31ZGO 89996108 Ki = 0.084 nM T74977 CX40VB 90000601 Ki = 3.7 nM T74977 C4W7YE 90000636 Ki = 3.3 nM T74977 C59PEY 90000723 IC50 = 62 nM T74977 C1EU3L 90000938 Ki = 0.78 nM T74977 CVU8R0 90176070 IC50 = 24 nM T74977 CK84DH 90176072 IC50 = 230 nM T74977 CW8NS3 90176086 IC50 = 1700 nM T74977 CE9SV3 90176089 IC50 = 14 nM T74977 CHU48V 90176101 IC50 = 2.3 nM T74977 C42HCL 90176105 IC50 = 2.6 nM T74977 C65DIN 90176117 IC50 = 9 nM T74977 C63ZAP 90176119 IC50 = 0.4 nM T74977 CS02UF 90176121 IC50 = 2.6 nM T74977 CM0SC1 90176154 IC50 = 2.5 nM T74977 CPY5V3 90176157 IC50 = 2.4 nM T74977 CM07CA 90176172 IC50 = 1.7 nM T74977 C28TDS 90176179 IC50 = 15 nM T74977 CB9Z3Y 90176183 IC50 = 2000 nM T74977 C7R8VF 90176191 IC50 = 1.8 nM T74977 CD2NL1 90176196 IC50 = 3 nM T74977 CT9F1Q 90176199 IC50 = 3.2 nM T74977 CDS1P5 90176200 IC50 = 7 nM T74977 CS0TW4 90176227 IC50 = 11 nM T74977 CRT7K1 91667406 Ki = 94700 nM T74977 CB5GU0 91668530 IC50 = 20 nM T74977 CSKI46 91885443 IC50 = 50 nM T74977 C64SIO 92042864 IC50 = 49 nM T74977 CGB54P 101902999 EC50 = 420 nM T74977 CG62HP 101903000 EC50 = 520 nM T74977 CSD75R 110868446 Ki > 100000 nM T74977 C7ML9C 110868449 Ki = 24800 nM T74977 CQ2C1F 117751256 IC50 = 4.8 nM T74977 C4QN9K 117751334 IC50 = 2 nM T74977 CHQJ26 117751337 IC50 = 4.6 nM T74977 CS2A6Q 117751339 IC50 = 2 nM T74977 CJB47R 118086034 Ki = 0.1 nM T74977 C71SUY 118348977 Ki = 0.11 nM T74977 C85WZU 118348985 Ki = 0.82 nM T74977 CE69MH 118349012 Ki = 0.088 nM T74977 CRSU68 118349055 Ki = 0.12 nM T74977 CY0K6A 118452766 IC50 = 2.2 nM T74977 C8JWK9 118452767 IC50 = 10 nM T74977 CHS4G0 118452789 IC50 = 4.9 nM T74977 C9KVQ0 118452843 IC50 = 2 nM T74977 C86XOE 118452846 IC50 = 7 nM T74977 C4FZ8M 118452870 IC50 = 21 nM T74977 CPZ0L6 118458718 IC50 = 2.2 nM T74977 CT06MH 118458775 IC50 = 13 nM T74977 C6AMJ8 118458786 IC50 = 1.1 nM T74977 CK6Z8O 118475621 IC50 = 180 nM T74977 CIVS69 118475644 IC50 = 143 nM T74977 C17FYA 118475649 IC50 = 355 nM T74977 CE49ZI 118475652 IC50 = 212 nM T74977 C0A9RJ 118475705 IC50 = 28.6 nM T74977 CKF24V 118712905 IC50 = 1800 nM T74977 CDHV30 118712906 IC50 = 18000 nM T74977 C8K6AY 118712907 IC50 = 17000 nM T74977 CZP0B9 118712908 IC50 > 50000 nM T74977 C01IKV 118712909 IC50 = 1400 nM T74977 CVFC04 118712910 IC50 = 5400 nM T74977 CRE4Z5 118712911 IC50 = 2300 nM T74977 CDT3W5 118712912 IC50 = 18000 nM T74977 CBR0O1 118712913 IC50 = 4300 nM T74977 CD0LS4 118712914 IC50 = 11000 nM T74977 C5O6GJ 118712915 IC50 = 330 nM T74977 CWE0S1 118712916 IC50 > 50000 nM T74977 CM6OV0 118712917 IC50 = 710 nM T74977 CY2LR5 118712918 IC50 > 5000 nM T74977 CR18YB 118712919 IC50 = 58 nM T74977 C63RXI 118712920 IC50 = 35 nM T74977 C95ABZ 118712921 IC50 = 24 nM T74977 C3FGD7 118712922 IC50 = 46 nM T74977 CW80GS 118713007 IC50 = 370 nM T74977 C61IJM 118732113 IC50 = 180 nM T74977 C3R0AG 118732114 IC50 = 460 nM T74977 C6EW5P 118732115 IC50 = 2500 nM T74977 C7IJW3 118732116 IC50 = 69 nM T74977 C7P5DG 118732117 IC50 = 490 nM T74977 C2PHU7 118732118 IC50 = 8.5 nM T74977 C1GSU3 118732119 IC50 = 6.6 nM T74977 CMFR46 118732120 IC50 = 1.3 nM T74977 CGCU39 118732121 IC50 = 6.8 nM T74977 C8ID7P 118732122 IC50 = 5.6 nM T74977 C2Y7NP 118732123 IC50 = 6.6 nM T74977 CUFI51 118732124 IC50 = 0.3 nM T74977 C1E4LP 118732125 IC50 = 13 nM T74977 CEN4F3 118732126 IC50 = 4.2 nM T74977 C5G1RM 118732127 IC50 = 5.5 nM T74977 CQSF74 118735386 IC50 = 3 nM T74977 C2P7NL 118735389 IC50 = 1.2 nM T74977 C5HSK4 118735401 IC50 = 13 nM T74977 C7XBQ8 119025602 IC50 = 810 nM T74977 CB94ME 119025603 IC50 = 46 nM T74977 CV0ZL6 121320413 IC50 = 3420 nM T74977 CG9Q1H 121320416 IC50 = 356 nM T74977 C4WY9G 121320420 IC50 = 13152 nM T74977 CRH42C 124124034 Ki = 0.047 nM T74977 C4CX9Y 124124085 Ki = 0.2 nM T74977 C2V8JF 124124180 Ki = 4 nM T74977 C0KD4B 127044233 IC50 = 140 nM T74977 C0B7QU 127048362 IC50 = 32 nM T74977 CX8W4F 127049041 IC50 = 0.7 nM T74977 CK5GJ2 127052461 IC50 = 0.94 nM T74977 CTG4P2 130289079 IC50 = 2.7 nM T74977 C9FUK2 135151360 IC50 = 5011.87 nM T74977 CHA4N2 136013680 IC50 > 10 nM T74977 CZ7EX0 136183413 IC50 = 8750 nM T74977 C1YUD0 136219394 IC50 > 10 nM T74977 CIU8W3 136254389 IC50 > 10 nM T74977 CZ9BN4 138320062 IC50 = 0.7 nM T74977 C4V1GH 145714280 IC50 = 39.81 nM T74977 C8RN4T 145979750 Ki = 11000 nM T74977 C6SM4I 145980334 Ki = 367300 nM T74977 C6IY7Q 145984119 Ki = 0.38 nM T74977 CYGF41 145985370 Ki = 0.19 nM T74977 CS19XQ 145985708 Ki = 0.12 nM T74977 C93FZG 145988498 Ki = 3200 nM T74977 CZ6IP8 145989872 Ki = 30100 nM T74977 CKT7O3 145993958 Ki = 269300 nM T74977 CNSJ07 155511845 Ki < 0.5 nM T74977 C2MD1Q 155513187 IC50 > 10000 nM T74977 C0KI2X 155517513 IC50 = 2.2 nM T74977 C5A1FL 155521427 Ki < 0.5 nM T74977 CC7W1O 155521798 IC50 = 0.6 nM T74977 CI6C9E 155532159 IC50 = 3.2 nM T74977 C31QWU 155536065 IC50 = 1 nM T74977 CP25WZ 155539880 IC50 = 19.95 nM T74977 CYT7A6 155542526 IC50 = 16 nM T74977 CP6ZS5 155545935 IC50 = 1.3 nM T74977 CPW73Q 155550391 IC50 = 2.5 nM T74977 C7QW1A 155553543 IC50 = 7.2 nM T74977 CVQ20P 155554448 IC50 = 1 nM T74977 C7BYX6 155562324 IC50 = 1.3 nM T74977 D00JMT 210332 IC50 = 2.8 nM T74977 D02PVB 8515 IC50 = 98 nM T74977 D08HFG 24809764 IC50 > 10000 nM T74977 D09HVH 135566652 IC50 > 10 nM T74977 D0UO2H 44556162 IC50 = 8 nM T65266 D09ZZW 503536 IC50 = 1500 nM T65266 C6IQV0 482174 IC50 = 5700 nM T65266 CY61LO 487910 IC50 = 1700 nM T65266 C6K5JV 487911 IC50 = 16000 nM T65266 C3J5VH 487912 IC50 = 1000 nM T65266 CZNK70 487918 IC50 = 330 nM T65266 CDN3F2 487919 IC50 = 1630 nM T65266 CT76XW 487920 IC50 = 2100 nM T65266 CVA82G 487921 IC50 = 460 nM T65266 CBR46W 487922 IC50 = 1400 nM T65266 CAJ64Q 490750 IC50 < 1000 nM T65266 CMO49H 491114 IC50 = 4300 nM T65266 COB17R 492544 IC50 > 50000 nM T65266 C68MZE 492548 IC50 > 100000 nM T65266 C4JO9E 492549 IC50 = 3280 nM T65266 C1JEY2 492550 IC50 = 300 nM T65266 CRML27 492552 IC50 = 380 nM T65266 C84QRW 493418 IC50 = 5700 nM T65266 CY1WF7 497453 IC50 = 3000 nM T65266 C43PXV 503499 IC50 = 2400 nM T65266 C2BSI5 503516 IC50 = 14000 nM T65266 CFRT87 503517 IC50 = 5400 nM T65266 C3JB0U 503520 IC50 = 13000 nM T65266 CA72XJ 503521 IC50 = 5200 nM T65266 CF14KO 503522 IC50 = 7400 nM T65266 CH18YP 503523 IC50 = 4600 nM T65266 CG6T1D 503524 IC50 = 4100 nM T65266 CLY7T8 503525 IC50 = 750 nM T65266 C37MIA 503526 IC50 = 1000 nM T65266 C8U2AD 503527 IC50 = 12000 nM T65266 CO6R4G 503528 IC50 = 2000 nM T65266 CHA5F8 503529 IC50 > 50000 nM T65266 C41DVG 503530 IC50 = 21000 nM T65266 C5XRJ6 503531 IC50 = 1200 nM T65266 CI1V6W 503532 IC50 > 50000 nM T65266 C84DXH 503533 IC50 = 1400 nM T65266 C7R3CM 503534 IC50 = 2000 nM T65266 CCMU16 503535 IC50 = 3000 nM T65266 C1E4IO 504181 IC50 = 2700 nM T65266 CEJ6U1 504182 IC50 = 1800 nM T65266 CZDS90 504183 IC50 = 1600 nM T65266 C04ONL 504184 IC50 = 2200 nM T65266 C65XPH 504185 IC50 = 11000 nM T65266 CRZN68 504186 IC50 = 42000 nM T65266 CK8CA2 504187 IC50 > 60000 nM T65266 C01MYV 504188 IC50 = 5800 nM T65266 C4C5WD 504189 IC50 = 4300 nM T65266 CIB52E 504190 IC50 = 230 nM T65266 CQ6L1G 504191 IC50 = 12000 nM T65266 C4CW5A 504192 IC50 > 60000 nM T65266 C09ACU 504193 IC50 > 60000 nM T65266 C7T0AD 504194 IC50 = 1300 nM T65266 C7VZY1 504195 IC50 > 60000 nM T65266 CU4EK0 504196 IC50 = 3600 nM T65266 COUS53 504197 IC50 = 5300 nM T65266 CTE3B4 504198 IC50 = 7700 nM T65266 CT81MP 504676 IC50 = 3500 nM T65266 C9FI5K 504680 IC50 = 10600 nM T65266 C8IFN4 504681 IC50 = 31000 nM T65266 CV6OY3 506523 IC50 = 1400 nM T65266 CQX7S4 506524 IC50 = 390 nM T65266 CXD73I 506525 IC50 = 1800 nM T65266 C6ANI5 506528 IC50 = 9000 nM T65266 CRU30I 507613 IC50 = 900 nM T65266 CI8SQ4 511361 IC50 > 50000 nM T65266 C02LPN 511362 IC50 = 30000 nM T65266 CJIW67 511363 IC50 = 13000 nM T65266 C3KG1M 511364 IC50 = 43000 nM T65266 CU85HK 511365 IC50 = 10700 nM T65266 C20EKN 511366 IC50 = 5900 nM T65266 C3FX8J 511367 IC50 = 31000 nM T65266 C4DEY1 511368 IC50 = 3700 nM T65266 CC2J9M 511369 IC50 = 5600 nM T65266 CIU5M2 511370 IC50 = 11000 nM T65266 C5CG4I 511371 IC50 = 5000 nM T65266 CTO87P 511372 IC50 = 2700 nM T65266 C5BJ6S 511373 IC50 = 26000 nM T65266 CDWB40 511374 IC50 = 15000 nM T65266 CDH29C 511375 IC50 = 31000 nM T65266 C8ZJD7 511376 IC50 = 31000 nM T65266 CJ56OH 513150 IC50 < 10000 nM T65266 C5BN4U 513891 IC50 = 12000 nM T65266 CVI54C 657065 IC50 = 1200 nM T65266 CUC54L 3008068 IC50 = 5000 nM T65266 CJ5NO6 3008069 IC50 = 34000 nM T65266 CQO9Y3 3008070 IC50 > 32000 nM T65266 CXM1K9 3008071 IC50 > 50000 nM T65266 CJ2NY3 3008418 IC50 = 20000 nM T65266 CIJ2T0 3008419 IC50 > 50000 nM T65266 CWD1X0 3008420 IC50 = 14000 nM T65266 C4K2JP 3008421 IC50 > 50000 nM T65266 CAN83S 3008422 IC50 = 13000 nM T65266 CMDQ27 4468931 IC50 = 1800 nM T65266 CK9WY1 5278824 IC50 = 100 nM T65266 C5MEQ4 5278825 IC50 = 110 nM T65266 C1F0AN 5278826 IC50 = 45 nM T65266 CV0O6S 5482516 IC50 = 15600 nM T65266 CEM30Z 5483089 IC50 = 8900 nM T65266 CJL21S 9853197 IC50 = 60 nM T65266 CJW4M9 9917616 IC50 = 11000 nM T65266 C39ZBC 10207572 IC50 = 30000 nM T65266 CGA86Z 10259200 IC50 = 12000 nM T65266 CJ46UK 10439772 IC50 = 420 nM T65266 COM8C5 21148125 IC50 = 16000 nM T65266 C1TW3V 22209806 IC50 > 50000 nM T65266 C8GVX3 22209808 IC50 > 50000 nM T65266 C6AS7E 22209811 IC50 = 3300 nM T65266 CLW13P 22209812 IC50 = 1700 nM T65266 C1TA6Z 22209813 IC50 = 440 nM T65266 CGUC83 22210989 IC50 = 58000 nM T65266 CV97ER 22210996 IC50 = 18000 nM T65266 C2BA1K 22211000 IC50 = 27000 nM T65266 C78AKX 22211010 IC50 > 100000 nM T65266 CL7M9B 22211011 IC50 = 32000 nM T65266 C1L8TE 22211012 IC50 = 18000 nM T65266 C0NYS5 22211016 IC50 = 50000 nM T65266 C67QJW 22211018 IC50 > 100000 nM T65266 CV9S2O 22211019 IC50 = 13000 nM T65266 C4UB6Q 22211020 IC50 = 14000 nM T65266 CBUV46 22211021 IC50 = 62000 nM T65266 CS9B7N 22211022 IC50 > 100000 nM T65266 CK81WO 25078062 IC50 = 3400 nM T65266 CYDW71 44268661 IC50 > 60000 nM T65266 C6S3AT 44268682 IC50 > 60000 nM T65266 CDJ0X4 44308299 IC50 > 100000 nM T65266 CIO1C2 44308345 IC50 > 100000 nM T65266 CX14BI 44308422 IC50 > 100000 nM T65266 CE3PS8 44308752 IC50 = 34000 nM T65266 CK2P5O 44375061 IC50 > 50000 nM T65266 C4CVW1 44375110 IC50 > 50000 nM T65266 C72KUL 44375154 IC50 = 9400 nM T65266 C1SBO9 44375192 IC50 > 50000 nM T65266 C42GUE 44375229 IC50 = 5300 nM T65266 CX76FI 44388198 IC50 = 350 nM T65266 CVW6O4 44399745 IC50 = 79432.82 nM T65266 CDRP83 44399750 IC50 = 50118.72 nM T65266 CW6NY8 44399751 IC50 = 5011.87 nM T65266 CM5W8Q 44399752 IC50 = 6309.57 nM T65266 C34WSP 44399753 IC50 = 10000 nM T65266 CE0T1O 44399754 IC50 = 1995.26 nM T65266 CT86CR 44399784 IC50 = 25118.86 nM T65266 C6GWS9 44399837 IC50 = 31622.78 nM T65266 C4AI1T 44399861 IC50 = 100000 nM T65266 CTX79F 44399866 IC50 = 25118.86 nM T65266 CP4KB7 44399867 IC50 = 794.33 nM T65266 C0WRU5 44399868 IC50 = 15848.93 nM T65266 C8JP2A 44399889 IC50 = 50118.72 nM T65266 CO4H3V 44399938 IC50 = 10000 nM T65266 CYH7F9 44399975 IC50 = 6309.57 nM T65266 CZRF38 44399976 IC50 = 6309.57 nM T65266 CATH48 44399977 IC50 = 6309.57 nM T65266 CL9NS3 44399978 IC50 > 199526.23 nM T65266 C9YO4K 44399979 IC50 > 199526.23 nM T65266 CX8M3O 44400003 IC50 = 39810.72 nM T65266 C4X1OG 44400004 IC50 = 19952.62 nM T65266 C5EV1S 44400005 IC50 = 158489.32 nM T65266 CFRU27 44400006 IC50 = 199526.23 nM T65266 C7FO3T 44400007 IC50 = 251188.64 nM T65266 CA6P2U 44400008 IC50 = 100000 nM T65266 CQP47M 44400009 IC50 = 7943.28 nM T65266 CCRB97 44400010 IC50 = 3981.07 nM T65266 CT40SR 44400033 IC50 = 31622.78 nM T65266 CA96HO 44400076 IC50 > 1000000 nM T65266 CX7O2Z 44400112 IC50 > 199526.23 nM T65266 C6Z5NC 44400113 IC50 > 199526.23 nM T65266 C6PCE5 44400114 IC50 = 31622.78 nM T65266 C95CRD 44400115 IC50 = 19952.62 nM T65266 CW5G3Z 73347065 IC50 > 50000 nM T65266 C6TNQ8 135412361 IC50 = 800 nM T65266 C53AWL 135434400 IC50 = 100 nM T83009 D0AZ3C 5291 IC50 = 272 nM T83009 D0OB0F 5328940 IC50 = 0.5 nM T83009 D0E3TC 44259 IC50 = 15.8 nM T83009 D03BNU 59604787 IC50 > 10000 nM T83009 D0T3ME 156422 IC50 > 30000 nM T83009 C9TU1O 16046126 IC50 > 1000 nM T83009 CURN06 24826798 IC50 = 39 nM T83009 C3VRO9 44557921 IC50 > 10000 nM T83009 CY90BD 49818230 IC50 = 685 nM T83009 CD2K4R 50908681 Ki > 1000000 nM T83009 C8NA4L 53384644 IC50 > 30000 nM T83009 C8AB1J 54759606 Ki = 180 nM T83009 CI50KU 58167984 IC50 = 863 nM T83009 CV63UL 67240318 IC50 > 10000 nM T83009 CRC5M0 71605046 IC50 = 11 nM T83009 C7GN8S 71605048 IC50 = 10 nM T83009 CT90RH 71605222 IC50 = 6 nM T83009 CBW27Q 71605223 IC50 = 298 nM T83009 C64OFJ 71605224 IC50 = 12 nM T83009 C4ZHD2 71605225 IC50 = 66 nM T83009 CEL6H2 71605226 IC50 = 36 nM T83009 C3CB5M 71605407 IC50 = 18 nM T83009 C3YL2D 71605408 IC50 = 40 nM T83009 CPG3A5 86302574 IC50 > 30000 nM T83009 C4X7SD 122192466 IC50 > 10000 nM T83009 CXC69T 137321158 IC50 = 306 nM T83009 C2MD1Q 155513187 IC50 > 10000 nM T83009 C8H1CZ 155536201 IC50 = 540 nM T83009 D0JR3W 71605047 IC50 = 2 nM T10897 D0S0RS 24988881 IC50 = 1 nM T10897 C3DCR6 890653 IC50 = 1400 nM T10897 C9O1HG 1113594 IC50 = 3 nM T10897 C3OW0E 9151192 IC50 = 1218 nM T10897 C2W4HU 11155946 IC50 = 5870 nM T10897 CO64DQ 11178786 IC50 = 66 nM T10897 C7HQ9V 11178995 IC50 = 100 nM T10897 C4R2VQ 11202128 IC50 = 24 nM T10897 CW34YK 11225042 IC50 = 6400 nM T10897 CCE6Z8 11271611 IC50 = 18 nM T10897 C3VD1K 11351351 IC50 = 2400 nM T10897 C5LOG6 11374374 IC50 = 62 nM T10897 CRV4N3 11375090 IC50 = 250 nM T10897 C9FV4H 11408261 IC50 = 101 nM T10897 C2ED6J 11430525 IC50 = 290 nM T10897 C1LP9U 11442719 IC50 = 119 nM T10897 CR29HU 11453250 IC50 = 192 nM T10897 C7JR4H 11487680 IC50 = 39 nM T10897 C5G2OA 11488029 IC50 = 10 nM T10897 CEFZ78 11670502 IC50 = 23 nM T10897 CT5L7H 11698083 IC50 = 28 nM T10897 C8J5NP 15980638 IC50 = 1 nM T10897 C2GVL4 15980639 IC50 > 50000 nM T10897 C1VQZ8 15980754 IC50 = 39 nM T10897 CG29FR 16034999 IC50 = 70 nM T10897 CN72LH 16035003 IC50 = 3 nM T10897 CZON96 16035660 IC50 = 9 nM T10897 C71BHJ 16035762 IC50 = 125 nM T10897 CKA78M 16035765 IC50 = 37 nM T10897 CJ71FD 16035876 IC50 = 12 nM T10897 C13RAO 16042458 IC50 = 21 nM T10897 CUD5R1 16732433 IC50 = 670 nM T10897 C5KS7D 17753032 IC50 = 30 nM T10897 CIJ73Z 24178407 IC50 = 48 nM T10897 CK7CA3 24573092 IC50 = 915 nM T10897 CMCJ08 24573104 IC50 = 145 nM T10897 CUQB24 24771823 IC50 = 2412 nM T10897 C20DOR 24829557 IC50 = 3.2 nM T10897 C0T3JN 24829559 IC50 = 15 nM T10897 C6F8WK 24829560 IC50 = 13 nM T10897 CED2J1 24829724 IC50 = 120 nM T10897 CZ1L2O 24830061 IC50 = 16 nM T10897 C6GFI1 24830062 IC50 = 2.8 nM T10897 CV4ZE1 24830229 IC50 = 120 nM T10897 CQX6Z4 24830385 IC50 = 81 nM T10897 CG07TH 24830387 IC50 = 100 nM T10897 CARS57 24830388 IC50 = 47 nM T10897 C7K2YC 24830389 IC50 = 47 nM T10897 C7IGH8 24830545 IC50 = 2500 nM T10897 C1J7DS 24830549 IC50 = 51 nM T10897 C7ING1 24830704 IC50 = 16 nM T10897 CK5B4V 24831014 IC50 = 96 nM T10897 C1UCN9 24831015 IC50 = 210 nM T10897 CGIJ84 24831655 IC50 = 21 nM T10897 C3NO5W 24831821 IC50 = 40 nM T10897 C9S1AO 24831822 IC50 = 34 nM T10897 C2HZ9D 24831825 IC50 = 8.6 nM T10897 C75ZOE 24831991 IC50 = 3.3 nM T10897 CMGN79 24831992 IC50 = 13 nM T10897 C1FZS6 24855892 IC50 = 257 nM T10897 CIL78S 24881032 IC50 = 268 nM T10897 CQ2T0G 24954326 IC50 = 618 nM T10897 CYB47H 24957857 IC50 = 675 nM T10897 C49JFY 24962977 IC50 = 9983 nM T10897 C3Y5NT 24970324 IC50 = 9 nM T10897 CF72XG 24970336 IC50 = 410 nM T10897 CN1A6D 24983658 IC50 = 26 nM T10897 C3W4YV 24983663 IC50 = 1510 nM T10897 C3P9OY 24984128 IC50 = 50 nM T10897 CZ65OP 24984927 IC50 = 2578 nM T10897 C0C6RI 24985101 IC50 = 61 nM T10897 CPIR62 24985271 IC50 = 2536 nM T10897 CX28KD 24988880 IC50 = 904 nM T10897 CP0L6U 24989358 IC50 = 100 nM T10897 CLB24O 24989744 IC50 = 99 nM T10897 C4C0PX 25016055 IC50 = 1 nM T10897 C0HGC5 25016056 IC50 = 4 nM T10897 CIC73W 25016057 IC50 = 7 nM T10897 C6NX7Z 25016310 IC50 = 6 nM T10897 CP13LW 25016311 IC50 = 0.3 nM T10897 CY1FJ7 25016312 IC50 = 1 nM T10897 CET01M 25016313 IC50 = 1 nM T10897 C8JV4R 25016314 IC50 = 0.45 nM T10897 C6YJ7T 25016566 IC50 = 0.03 nM T10897 CS63KE 25065534 IC50 = 7 nM T10897 CPX6J7 25065739 IC50 = 780 nM T10897 COE54Z 25065742 IC50 = 4466 nM T10897 C48SFQ 25093806 IC50 = 250 nM T10897 C68CBZ 25093881 IC50 = 1670 nM T10897 C0LQ6Z 25094160 IC50 > 3000 nM T10897 CDB4Q8 25094198 IC50 = 4000 nM T10897 CM5F1B 25094199 IC50 = 4600 nM T10897 C7JPL0 25094597 IC50 = 53 nM T10897 CWBY02 25094599 IC50 = 194 nM T10897 CSKV62 25094874 IC50 = 2175 nM T10897 C1X2OV 25094875 IC50 = 158 nM T10897 CZ9J6X 25094877 IC50 = 63 nM T10897 CN9FP8 25095149 IC50 = 10 nM T10897 C3QDS9 25095675 IC50 = 140 nM T10897 C3HG8F 25095930 IC50 = 398 nM T10897 CRF62S 25096446 IC50 = 9 nM T10897 C9FH5C 25099088 IC50 = 4 nM T10897 CF7ON5 25099235 IC50 = 8.8 nM T10897 CLQR14 25099433 IC50 = 6.7 nM T10897 CWG03M 25099435 IC50 = 4.8 nM T10897 CJS08Y 25115386 IC50 = 0.04 nM T10897 CV7S8R 25121742 IC50 = 8.1 nM T10897 C1BJ8R 25121743 IC50 = 4.2 nM T10897 CE4Q6L 25121744 IC50 = 3.8 nM T10897 C9ZCL8 25121745 IC50 = 5.2 nM T10897 CDS2W1 25122095 IC50 = 6.3 nM T10897 C89TQD 25122096 IC50 = 3.2 nM T10897 C9AJ6Q 25122097 IC50 = 3.8 nM T10897 CLK5J6 25122467 IC50 = 8.7 nM T10897 CPD5E2 25155079 IC50 > 1000 nM T10897 CWY50V 25155343 IC50 = 68 nM T10897 CE5A1G 25157288 IC50 = 193 nM T10897 CRHL29 25157290 IC50 = 250 nM T10897 CCYQ62 25157578 IC50 = 220 nM T10897 C2WMH9 25158453 IC50 = 119 nM T10897 CH3M0T 25158717 IC50 = 180 nM T10897 C3F5EO 25159235 IC50 = 79 nM T10897 C5EJ9L 25159237 IC50 = 110 nM T10897 CV6UH1 25167051 IC50 = 41 nM T10897 C1W0CN 25167053 IC50 = 3870 nM T10897 CTG6R0 25167056 IC50 > 40000 nM T10897 CUP3X7 25167252 IC50 > 40000 nM T10897 CGDC51 25172945 IC50 = 28 nM T10897 C19AXU 25175138 IC50 = 313 nM T10897 CCE3F0 25192354 IC50 = 2340 nM T10897 CD0SE6 25192355 IC50 = 1360 nM T10897 CXL4I2 25192356 IC50 = 1160 nM T10897 CYHO16 25192357 IC50 = 439 nM T10897 C1EFN8 25192358 IC50 = 179 nM T10897 CYE52U 25192509 IC50 = 157 nM T10897 CWI3V4 25204855 IC50 = 53 nM T10897 CN6D5T 25204857 IC50 = 168 nM T10897 C79PEH 42601472 IC50 = 0.05 nM T10897 CK9D4B 44192371 IC50 = 66 nM T10897 CAOM13 44193601 IC50 = 945 nM T10897 CE76IQ 44247738 IC50 = 27 nM T10897 C3CKN7 44250031 IC50 = 3 nM T10897 C6RM7N 44425923 IC50 = 580 nM T10897 CY26TW 44425926 IC50 = 560 nM T10897 CG3M9Q 44425928 IC50 = 140 nM T10897 CY17AF 44425929 IC50 = 7300 nM T10897 C3RM8B 44425930 IC50 > 1000 nM T10897 C9ZK3W 44425932 IC50 = 90 nM T10897 C4T2NF 44425934 IC50 = 97 nM T10897 C61FVA 44425935 IC50 = 110 nM T10897 C7ZS3J 44425936 IC50 = 390 nM T10897 C7KBV1 44425938 IC50 = 120 nM T10897 C9F8TS 44425939 IC50 = 430 nM T10897 CXDA73 44425940 IC50 = 350 nM T10897 CRY87K 44425941 IC50 = 780 nM T10897 C7UT1J 44425942 IC50 > 10000 nM T10897 CAEG93 44425943 IC50 > 10000 nM T10897 C1XF3Y 44425944 IC50 = 94 nM T10897 COWA07 44425945 IC50 = 51 nM T10897 CPD97U 44425946 IC50 = 39 nM T10897 CIOC38 44425950 IC50 = 260 nM T10897 CEQH83 44425952 IC50 = 100 nM T10897 CK63OU 44425954 IC50 = 110 nM T10897 CGHV69 44425956 IC50 = 99 nM T10897 C1PKM9 44425958 IC50 = 110 nM T10897 CQCY18 44425959 IC50 = 550 nM T10897 C8L0EY 44425962 IC50 = 39 nM T10897 C4YCL8 44425964 IC50 = 210 nM T10897 CIO54U 44425965 IC50 = 340 nM T10897 CK4R8X 44425966 IC50 = 6300 nM T10897 C56XKL 44425969 IC50 = 58 nM T10897 C2H9SM 44425971 IC50 = 38 nM T10897 CNC37Y 44425972 IC50 = 51 nM T10897 CW6F1B 44425975 IC50 = 470 nM T10897 CG5XL8 44425978 IC50 = 35 nM T10897 CCV7B9 44425980 IC50 = 100 nM T10897 CPL5N6 44425982 IC50 > 1000 nM T10897 CNU3S9 44464942 IC50 = 24 nM T10897 CHX91U 44465204 IC50 = 30 nM T10897 CH82YS 44465209 IC50 = 342 nM T10897 CPFD18 44465469 IC50 = 15 nM T10897 C3RJ8W 44465470 IC50 = 231 nM T10897 C48FES 44465471 IC50 = 1705 nM T10897 CM7E3U 44465474 IC50 = 113 nM T10897 CF6H9G 44465737 IC50 = 19 nM T10897 C8M5RP 44468455 IC50 = 68 nM T10897 CWNA17 44470234 IC50 = 13 nM T10897 C65WRK 44470235 IC50 = 130 nM T10897 C1PW9T 44470237 IC50 = 3.1 nM T10897 C8D5WB 44513582 IC50 = 0.5 nM T10897 CE0OJ6 44573270 IC50 = 180 nM T10897 C0Q7YV 44573583 IC50 = 6.5 nM T10897 CP40XE 44573664 IC50 = 140 nM T10897 CO53TY 44573709 IC50 = 5.6 nM T10897 CRC34F 44573710 IC50 = 36 nM T10897 C91BFS 44573711 IC50 = 92 nM T10897 CL1EV5 44573749 IC50 = 9.6 nM T10897 C16CEN 44573750 IC50 = 110 nM T10897 C7DP5H 44574621 IC50 = 1150 nM T10897 C6YUF7 44574659 IC50 = 790 nM T10897 CXHU46 44574733 IC50 = 49 nM T10897 C76MCZ 44574768 IC50 > 1000 nM T10897 C9U2HK 44602491 IC50 = 2 nM T10897 CH53BJ 45267253 IC50 = 145 nM T10897 CQ06MG 45267479 IC50 = 59 nM T10897 CQ9DI7 45267552 IC50 = 9 nM T10897 C5I3DF 45267558 IC50 = 10 nM T10897 CKHB14 45268123 IC50 > 1000 nM T10897 CEM01Y 45268125 IC50 = 32 nM T10897 C8VWD5 45268354 IC50 = 82 nM T10897 CF0VD5 45269006 IC50 > 9999 nM T10897 CD18NK 45269011 IC50 = 15 nM T10897 CB81XL 45269205 IC50 = 4 nM T10897 CVO1X0 45269289 IC50 > 9999 nM T10897 CD1P7C 45269851 IC50 = 32 nM T10897 CPA0R2 45269854 IC50 = 884 nM T10897 COF39V 45269859 IC50 = 16 nM T10897 CH50LG 45270080 IC50 = 13 nM T10897 CFJR23 45270133 IC50 = 1402 nM T10897 CW91FD 45270672 IC50 = 8 nM T10897 C2I7UW 45270677 IC50 = 828 nM T10897 CIW1C9 45270685 IC50 = 0.6 nM T10897 CB5HN1 45270695 IC50 = 12 nM T10897 CRKY53 45270906 IC50 = 2.9 nM T10897 C2NH1L 45271744 IC50 = 1 nM T10897 CC87PO 45271819 IC50 > 9999 nM T10897 CVJK74 45272403 IC50 = 0.2 nM T10897 C0VE1G 45272410 IC50 = 2 nM T10897 CV9Q2X 45272423 IC50 = 11 nM T10897 C1NZV4 45272613 IC50 = 2162 nM T10897 C01DJY 45272620 IC50 = 0.6 nM T10897 C6PH8O 45272625 IC50 = 9 nM T10897 COK58D 45272681 IC50 = 4377 nM T10897 C4FU1S 45273509 IC50 = 11 nM T10897 C37YCG 45273521 IC50 = 125 nM T10897 C6P7OK 45482159 IC50 > 1000 nM T10897 CV9L4M 45482167 IC50 = 2.7 nM T10897 CWQP02 45487280 IC50 = 68000 nM T10897 CTM2G3 45487353 IC50 = 4000 nM T10897 CBH5J7 45487394 IC50 = 13000 nM T10897 C3K6AE 46174454 IC50 > 100000 nM T10897 CYLJ13 46224621 IC50 = 25 nM T10897 CM3U2E 46224622 IC50 = 5 nM T10897 C3FYJ4 46224627 IC50 = 60 nM T10897 CMKB61 46224628 IC50 = 7 nM T10897 CD86TL 46224629 IC50 = 7 nM T10897 CY4WS0 46224632 IC50 = 80 nM T10897 C7S5OG 46224633 IC50 = 390 nM T10897 CM3W5X 46224637 IC50 = 311 nM T10897 CYLF47 46224638 IC50 = 22 nM T10897 C21FAC 46224648 IC50 = 7 nM T10897 CJ3V2S 46224650 IC50 = 10 nM T10897 C8SL1A 46224651 IC50 = 25 nM T10897 C6QAO5 46224655 IC50 = 820 nM T10897 C85WLX 46224656 IC50 = 187 nM T10897 CRQP47 46224660 IC50 = 108 nM T10897 CM87AT 46224663 IC50 = 11 nM T10897 C0Z6BJ 46226093 IC50 = 156 nM T10897 CX90QP 46226094 IC50 = 33 nM T10897 CWE8I5 46226134 IC50 = 6 nM T10897 C6DW5V 46226153 IC50 = 2 nM T10897 C9E6TW 46226154 IC50 = 10 nM T10897 CBX49E 46226155 IC50 = 1 nM T10897 C9MT5B 46226170 IC50 = 38 nM T10897 CNH40X 46226171 IC50 = 16 nM T10897 C90JXT 46226228 IC50 > 10000 nM T10897 C16JEA 46226230 IC50 = 20 nM T10897 CZ7XG8 46226241 IC50 > 10000 nM T10897 CI0HX5 46226243 IC50 = 0.69 nM T10897 CUCR36 46226244 IC50 = 230 nM T10897 CZNF54 46226259 IC50 = 16 nM T10897 C37ZLU 46226260 IC50 = 60 nM T10897 CX3WS4 46226261 IC50 = 49 nM T10897 CWBI12 46226262 IC50 = 61 nM T10897 CD60MT 46226279 IC50 = 0.068 nM T10897 C10UOF 46226280 IC50 = 76 nM T10897 CY1UH5 46226281 IC50 = 17 nM T10897 C2KV6Q 46871752 IC50 = 6308 nM T10897 C1KIM5 46880665 IC50 = 153 nM T10897 CI8M5H 46880666 IC50 = 24 nM T10897 C7B6DX 46880667 IC50 = 10 nM T10897 CLIK61 46880714 IC50 = 84 nM T10897 C8S2NW 46880716 IC50 = 6523 nM T10897 CP9MF7 46880717 IC50 = 7 nM T10897 CNQ8J9 46880718 IC50 = 199 nM T10897 C49IYR 46880762 IC50 = 2823 nM T10897 C3VCP8 46880763 IC50 = 14 nM T10897 CGR9T7 46880764 IC50 = 1019 nM T10897 CI9M8N 46880765 IC50 = 174 nM T10897 CQ3S9C 46880803 IC50 = 775 nM T10897 CJ4N1K 46880805 IC50 = 55 nM T10897 C0IPS4 46880806 IC50 = 65 nM T10897 CMO72R 46880840 IC50 = 16 nM T10897 CWIE20 46897105 IC50 = 4200 nM T10897 CL13XO 46916546 IC50 = 50900 nM T10897 CR84FK 46916547 IC50 > 100000 nM T10897 CP6K5Q 46916548 IC50 = 27 nM T10897 CPX94F 46916597 IC50 > 100000 nM T10897 C06OCV 46916599 IC50 = 15400 nM T10897 C98QUX 49845330 IC50 = 0.1 nM T10897 CE1H3B 49845331 IC50 = 0.2 nM T10897 CKF06P 51346899 IC50 = 217 nM T10897 C9QJ6K 52940674 IC50 = 1760 nM T10897 C0AO5Y 52940686 IC50 = 731 nM T10897 CN5AY7 52941877 IC50 = 74 nM T10897 CQDW50 52941887 IC50 = 4246 nM T10897 CE3HF8 52943508 IC50 = 1308 nM T10897 CT4B6A 52945516 IC50 > 20000 nM T10897 C58ULQ 52945533 IC50 = 255 nM T10897 C1BV9R 52945548 IC50 = 60 nM T10897 C8NW6U 52947125 IC50 = 27 nM T10897 CAVT17 52949620 IC50 = 96 nM T10897 C2XZ7K 52953418 IC50 = 10 nM T10897 CM5OV9 53231164 IC50 > 1000 nM T10897 CFJH63 53231165 IC50 > 1000 nM T10897 CN7RE5 53231166 IC50 = 280 nM T10897 CZ2WV1 53231167 IC50 = 700 nM T10897 CX12FW 53231263 IC50 = 100 nM T10897 CE7S6K 53231264 IC50 = 40 nM T10897 CMI8Q3 53231266 IC50 = 600 nM T10897 C7XTO6 53231373 IC50 > 1000 nM T10897 CUVC81 53321551 IC50 = 88 nM T10897 C9S6NM 53388366 IC50 = 12588 nM T10897 C8TS1P 54742333 IC50 = 137 nM T10897 CPM97D 54742334 IC50 = 1692 nM T10897 CFTH57 54742335 IC50 = 783 nM T10897 CSL5C0 54742336 IC50 = 121 nM T10897 CF9RM6 54742337 IC50 > 1000 nM T10897 C7XCD3 54742338 IC50 = 34 nM T10897 C3E1VP 54742339 IC50 = 30 nM T10897 CK72ZM 54753987 IC50 = 37749 nM T10897 CW4B9D 56661556 IC50 < 39 nM T10897 C4SOW7 56664975 IC50 = 182 nM T10897 CTKZ54 56668408 IC50 = 47 nM T10897 C2XM7B 56671917 IC50 = 10639 nM T10897 C31BWR 56675293 IC50 = 319 nM T10897 CY87HU 56675294 IC50 = 17 nM T10897 C40WHM 56678629 IC50 = 755 nM T10897 C0HZW6 56678630 IC50 = 162 nM T10897 COPY39 56835181 IC50 = 969 nM T10897 CC2QT9 57390832 IC50 = 6715 nM T10897 C2ND7G 57390963 IC50 = 18259 nM T10897 C7PI5V 57392606 IC50 > 100000 nM T10897 CZ2NH8 57392695 IC50 = 1113 nM T10897 C8QL2Y 57392742 IC50 = 5080 nM T10897 CBE67I 57394327 IC50 > 60000 nM T10897 CCF9O2 57394328 IC50 = 20500 nM T10897 C08FYU 57394401 IC50 > 10000 nM T10897 CY7LK2 57397740 IC50 = 2450 nM T10897 C3ADI8 57397981 IC50 > 20000 nM T10897 C8U6JQ 57398030 IC50 = 8264 nM T10897 C4QAE6 57399403 IC50 = 9140 nM T10897 C6H5MA 57399624 IC50 = 550 nM T10897 C9ZUF6 57400850 IC50 = 760 nM T10897 CS9A6Q 57401169 IC50 > 10000 nM T10897 CE8RW7 57401334 IC50 = 128 nM T10897 CKGC06 57403093 IC50 = 9422 nM T10897 CBOF90 57744441 IC50 = 458 nM T10897 CM13EJ 57744449 IC50 = 329 nM T10897 C0YG6W 57744453 IC50 = 48 nM T10897 CI8OQ5 57744454 IC50 = 12 nM T10897 CAHQ26 57744455 IC50 = 55 nM T10897 CUVA50 57744489 IC50 = 191 nM T10897 CC42IM 57919836 IC50 = 227 nM T10897 CFC5O8 57919896 IC50 = 67 nM T10897 CUO25R 57919923 IC50 = 306 nM T10897 C46EAL 57919928 IC50 = 125 nM T10897 CCV32N 58031443 IC50 = 55 nM T10897 C1GYS0 58031447 IC50 = 46 nM T10897 CKZ0Q2 59179717 IC50 = 1925 nM T10897 CQP80B 59369702 IC50 = 2677 nM T10897 C0V6UI 59481190 IC50 = 268 nM T10897 CXV5J3 59481192 IC50 = 214 nM T10897 COQ1G3 59481196 IC50 = 135 nM T10897 CPIO31 59481226 IC50 = 194 nM T10897 C6RSG4 59481229 IC50 = 656 nM T10897 COQ91T 59481233 IC50 = 9 nM T10897 CS1W9P 59481254 IC50 = 39 nM T10897 CWI97F 59481258 IC50 = 95 nM T10897 CI82LP 59481269 IC50 = 8 nM T10897 CSY18A 59481280 IC50 = 40 nM T10897 CL6CE1 59481285 IC50 = 105 nM T10897 CLG4O8 59481287 IC50 = 219 nM T10897 CVWP50 59481289 IC50 = 32 nM T10897 C5RI1U 59481293 IC50 = 504 nM T10897 CA1NJ7 59481303 IC50 = 524 nM T10897 CM10SR 59481307 IC50 = 8 nM T10897 C0XQ6Z 59481311 IC50 = 477 nM T10897 C2N9BE 59481312 IC50 = 748 nM T10897 CEC4K9 66849498 IC50 = 125 nM T10897 CRNP95 67011239 IC50 = 660 nM T10897 C0DK6H 67012215 IC50 = 24 nM T10897 CHG37E 67012400 IC50 = 1100 nM T10897 C68SFN 68495091 IC50 = 236 nM T10897 CG86ZV 68556493 IC50 = 6.5 nM T10897 COW29T 71521050 IC50 = 41 nM T10897 C6V1UL 71521153 IC50 = 2249 nM T10897 CO5SK4 71521154 IC50 = 325 nM T10897 C4S2KL 71521265 IC50 = 68 nM T10897 C46VOH 71521266 IC50 = 124 nM T10897 C8O7LG 71568068 IC50 = 295 nM T10897 C4AL0C 71571569 IC50 = 15 nM T10897 C5DBQ3 71585291 IC50 = 2 nM T10897 CTN2M4 71585295 IC50 = 25 nM T10897 CD2FJ1 76311098 IC50 = 51 nM T10897 CL3N7Y 76311099 IC50 = 9 nM T10897 CFS8V3 76311109 IC50 = 30 nM T10897 CY9R6J 76311110 IC50 = 41 nM T10897 CNF8C4 76314705 IC50 = 14 nM T10897 C0WGF1 76314706 IC50 = 30 nM T10897 C5R7XU 76314719 IC50 = 6 nM T10897 CT3UC6 76314720 IC50 = 11 nM T10897 CZ02DS 76314721 IC50 = 42 nM T10897 CC4KI6 76318277 IC50 = 8 nM T10897 C8NL2A 76318294 IC50 = 12 nM T10897 C4XNS5 76318295 IC50 = 28 nM T10897 CRC9K8 76321980 IC50 = 6 nM T10897 CB27LM 76321985 IC50 = 9 nM T10897 CJF6L1 76325599 IC50 = 390 nM T10897 C4KEQ5 76325600 IC50 = 4 nM T10897 C0EJK8 76325610 IC50 = 21 nM T10897 C8YTS4 76325611 IC50 = 12 nM T10897 CO6JL5 76325612 IC50 = 218 nM T10897 COT36C 76325613 IC50 = 241 nM T10897 C3G1TU 76329165 IC50 = 54 nM T10897 CQA71J 76329166 IC50 = 0.5 nM T10897 C6AZ9E 76329177 IC50 = 6 nM T10897 C5FDL1 76332839 IC50 = 23 nM T10897 C7CZ5R 76332840 IC50 = 11 nM T10897 CQB36E 76332841 IC50 = 72 nM T10897 C8D0BI 76332842 IC50 = 2 nM T10897 CZ1S4C 76332843 IC50 = 99 nM T10897 C0VAU9 76336449 IC50 = 3 nM T10897 C1DRW8 76336462 IC50 = 407 nM T10897 C4YS2T 91885562 IC50 = 2.5 nM T10897 CXF57S 124192332 IC50 = 20 nM T10897 C9A6HL 124192338 IC50 = 21 nM T10897 C0EV1F 124192339 IC50 = 4.7 nM T10897 CP3Y5V 124192351 IC50 = 80 nM T10897 CV3QT1 124192413 IC50 = 11 nM T10897 C7LQG8 124192420 IC50 = 27 nM T10897 C7OY1T 124192446 IC50 = 1.2 nM T10897 CT3B9Y 124192448 IC50 = 15 nM T10897 CO6M9X 124192480 IC50 = 110 nM T10897 CM4BO1 124192487 IC50 = 9.5 nM T10897 CD3OI1 124192489 IC50 = 38 nM T10897 C82PDZ 135410872 IC50 = 29 nM T10897 C7DJ8X 135771804 IC50 = 59 nM T10897 C39IRY 135771805 IC50 = 16 nM T10897 CR0B8U 135870301 IC50 = 2326 nM T10897 C9C2RP 135874482 IC50 = 378 nM T10897 CXS24V 135876079 IC50 = 24345 nM T10897 CI2ZY5 137633527 IC50 = 19740 nM T10897 CV2S8K 137639011 IC50 = 130 nM T10897 CSNA51 137646974 IC50 = 190 nM T10897 CV9X2F 137654711 IC50 = 220 nM T10897 C0ZM1J 137657767 IC50 = 2.3 nM T10897 CM7NY2 137660491 IC50 = 100 nM T10897 CA19ZQ 145485632 IC50 = 17 nM T10897 CR6U7C 145485656 IC50 = 9.7 nM T10897 CNJ63T 145485676 IC50 = 4.5 nM T10897 CUVG50 145485772 IC50 = 7.5 nM T10897 CR59UO 145485790 IC50 = 3.9 nM T10897 CQ3YF1 145485794 IC50 = 5.1 nM T10897 CQ3A4W 145486036 IC50 = 30 nM T10897 C3PW5S 145488904 IC50 = 260 nM T10897 COTS02 145488943 IC50 = 4.8 nM T10897 CVIC57 145488948 IC50 = 3600 nM T10897 CZWX24 145488956 IC50 = 4.1 nM T10897 CK6ZE8 145488958 IC50 = 31 nM T10897 CZ2VC3 145488971 IC50 = 3 nM T10897 CYPR21 145488977 IC50 = 22 nM T10897 CR1L5Z 145489008 IC50 = 6.4 nM T10897 CL7ND2 145489022 IC50 = 6.4 nM T10897 CE03YV 145489030 IC50 = 58 nM T10897 CM0J2W 145489062 IC50 = 150 nM T10897 CX5PO2 145489063 IC50 = 5.1 nM T10897 CD0X5J 145489065 IC50 = 4.3 nM T10897 CR9CI8 145489123 IC50 = 2.8 nM T10897 CIT78H 145489146 IC50 = 760 nM T10897 CJ70ZU 145489152 IC50 = 3 nM T10897 CAZR34 145489153 IC50 = 5.3 nM T10897 C2BP8F 145489177 IC50 = 310 nM T10897 CDY13E 145489195 IC50 = 46 nM T10897 CZ70AC 145489228 IC50 = 4.5 nM T10897 CO4KE8 145489238 IC50 = 13 nM T10897 C7T1XQ 145489240 IC50 = 18 nM T10897 CDR7E1 145489259 IC50 = 5.5 nM T10897 CTS46Y 145489260 IC50 = 9.2 nM T10897 C5H2MB 145489263 IC50 = 570 nM T10897 CY1OZ9 145489307 IC50 = 14 nM T10897 CD4O7F 145489314 IC50 = 2700 nM T10897 CN23TE 145489338 IC50 = 8.9 nM T10897 C1Z7QC 145489339 IC50 = 5.5 nM T10897 CP6V1L 145987660 IC50 = 95 nM T10897 CAK58X 145989605 IC50 > 10000 nM T10897 C1VX2E 145992173 IC50 = 2700 nM T10897 D0O3TT 11973722 IC50 = 254 nM T10897 D0O7DP 25195516 IC50 = 6.1 nM T33455 C7M6EW 10086927 Ki = 28 nM T33455 C1DE6J 10905077 Ki > 10000 nM T33455 C0RMF2 10913569 Ki = 29 nM T33455 C2I4EZ 11046863 Ki > 10000 nM T33455 CP1HU8 11089952 Ki = 320 nM T33455 CQR7D9 11761685 Ki > 10000 nM T33455 CSU3N6 44300647 Ki = 850 nM T33455 C98QCZ 44300715 Ki > 10000 nM T33455 C9W4DE 135404272 Ki = 58 nM T33455 CSP1B5 135405043 Ki = 9 nM T33455 CA2VJ0 135405225 Ki = 70 nM T33455 CX0BI7 135409801 Ki = 27 nM T33455 CMY40H 135432255 Ki > 10000 nM T33455 C1URN2 135437180 Ki = 140 nM T33455 C2FXY6 135450996 Ki = 44 nM T33455 CV6Y1F 135465667 Ki = 70 nM T33455 C9WM7S 135490873 Ki = 7.5 nM T33455 C7NVX9 135524557 Ki = 8 nM T33455 CM7X4F 135525102 Ki = 13 nM T33455 CS2UA6 135539040 Ki = 9.4 nM T33455 CBZX07 135543997 Ki = 5.6 nM T33455 C3TSW1 135987621 Ki = 38 nM T33455 CD81HQ 135987622 Ki = 32 nM T33455 CTQ4C9 135987623 Ki = 29 nM T33455 C38XNC 135987624 Ki = 130 nM T33455 CX8L0M 135987625 Ki = 60 nM T33455 CHQ60J 135987626 Ki = 62 nM T33455 C9I6TM 135987627 Ki = 31 nM T33455 CRK3U7 135987628 Ki = 32 nM T33455 C97FWS 135987629 Ki = 12 nM T33455 C0F3PA 135987630 Ki = 20 nM T33455 CH3PQ8 135987631 Ki = 110 nM T33455 C0KD6S 135987632 Ki = 32 nM T33455 CPC43Z 135987633 Ki = 110 nM T33455 CJ38IR 135987634 Ki = 24 nM T33455 CY08HC 135987635 Ki = 25 nM T33455 CKZ04W 135987636 Ki = 11 nM T33455 CCR03Y 135987637 Ki = 51 nM T33455 CHC9Y2 135987638 Ki = 32 nM T33455 C8OM9V 135987643 Ki = 11 nM T33455 C7Y6US 135987645 Ki = 18 nM T33455 CYB1L7 135987655 Ki = 100 nM T33455 CMQU68 135987656 Ki = 110 nM T33455 C0E5MS 135987658 Ki = 72 nM T86597 D02YNI 9936746 Ki = 5.4 nM T86597 D05ICT 132010322 Ki = 4.6 nM T86597 D07OFM 46943432 IC50 = 32.5 nM T86597 D0M2TS 71600087 Ki = 1 nM T86597 D0PH9I 118693659 Ki = 100 nM T86597 D0ZW4W 46907787 Ki = 12.5 nM T86597 D09SFV 3973 IC50 = 10300 nM T86597 C92EYR 1503595 IC50 = 30000 nM T86597 C8BZ9Y 5325760 IC50 = 34300 nM T86597 CIG94A 13953713 IC50 = 25118.86 nM T86597 CO6HM1 16480179 IC50 = 22000 nM T86597 C3UFS6 39791103 IC50 = 3000 nM T86597 C2P0IW 44243549 IC50 = 6000 nM T86597 C3VRO9 44557921 IC50 > 10000 nM T86597 C98BLM 49871817 IC50 = 16 nM T86597 CG3PR6 52912222 IC50 = 3.162 nM T86597 CBXV52 52932793 IC50 = 199.53 nM T86597 CJE59U 52932930 IC50 = 3162.28 nM T86597 CSZ2T6 52932933 IC50 = 12589.25 nM T86597 CN87IR 52933159 IC50 = 2511.89 nM T86597 CG6OL4 52933160 IC50 = 794.33 nM T86597 CP8Y9K 52933161 IC50 = 1995.26 nM T86597 CK8Z4P 52933165 IC50 = 15848.93 nM T86597 CKC17F 52933403 IC50 = 1584.89 nM T86597 CD08ZX 52933405 IC50 = 3162.28 nM T86597 C1T7VQ 52933407 IC50 = 2511.89 nM T86597 CO8VX9 52933655 IC50 = 3162.28 nM T86597 C6G7BE 52933893 IC50 = 2511.89 nM T86597 C7VN1E 52934039 IC50 = 1584.89 nM T86597 CUZE18 52934122 IC50 = 1995.26 nM T86597 CN16FE 52934128 IC50 = 2511.89 nM T86597 CTS13B 52934275 IC50 = 1584.89 nM T86597 CNOH36 52935183 IC50 = 398.11 nM T86597 CLRH53 52935478 IC50 = 1995.26 nM T86597 CJIB35 53054190 IC50 = 5200 nM T86597 C6V8YR 53054191 IC50 = 14000 nM T86597 C09HTR 53054200 IC50 = 1400 nM T86597 CUS8F7 53054236 IC50 = 4300 nM T86597 CX5QN4 53054237 IC50 = 13000 nM T86597 CD2TY9 53054238 IC50 = 11000 nM T86597 C47GAW 53054240 IC50 = 4900 nM T86597 CVH2G1 53054241 IC50 = 2400 nM T86597 CF9E2V 53054248 IC50 = 2000 nM T86597 CRWK92 53054249 IC50 = 6000 nM T86597 CSXI51 53054250 IC50 = 2500 nM T86597 CM12EL 53054251 IC50 = 2500 nM T86597 CY5L3J 53054252 IC50 = 3600 nM T86597 CWV76Y 53054258 IC50 = 900 nM T86597 CIU8P7 53054259 IC50 = 500 nM T86597 CVX3R0 53054274 IC50 = 3900 nM T86597 CB05OM 53054276 IC50 = 1700 nM T86597 CLR97U 53054289 IC50 = 1500 nM T86597 CJ6E2Q 53054291 IC50 = 4400 nM T86597 C1WSZ4 53054297 IC50 = 2200 nM T86597 C7A2XC 53054319 IC50 = 1800 nM T86597 C0J1EO 53054320 IC50 = 4700 nM T86597 CK68UF 53054321 IC50 = 1100 nM T86597 CJY5S2 53054322 IC50 = 4200 nM T86597 C1YW5L 53054324 IC50 = 1500 nM T86597 C8Q6WG 53054325 IC50 = 1100 nM T86597 CQEF28 53308655 IC50 = 28200 nM T86597 C9V5LX 53318989 IC50 = 160 nM T86597 CEK3X6 54757749 IC50 = 7400 nM T86597 C1D3WH 54757750 IC50 = 4200 nM T86597 C1DZ7Y 54757751 IC50 = 3300 nM T86597 C6W5OZ 54757752 IC50 = 2300 nM T86597 C1KWY4 54759170 IC50 = 2000 nM T86597 C7HK2C 56924692 IC50 = 1500 nM T86597 CX6SD9 56950289 IC50 = 3600 nM T86597 CZ6NE0 56950420 IC50 = 1500 nM T86597 CJ5BE9 56950421 IC50 = 3600 nM T86597 CL96VQ 56950422 IC50 = 1900 nM T86597 CCLD98 56950423 IC50 = 12000 nM T86597 CZD7G2 56950424 IC50 = 5600 nM T86597 CPQ0B7 56950425 IC50 = 8100 nM T86597 CL90DK 56950426 IC50 = 800 nM T86597 CF9IJ1 56950561 IC50 = 800 nM T86597 CH24QC 56950562 IC50 = 14000 nM T86597 CU62NO 56950563 IC50 = 16000 nM T86597 CRD86M 56950564 IC50 = 19000 nM T86597 CNQ2L5 56950565 IC50 = 31000 nM T86597 CB3A1Z 56950566 IC50 = 11000 nM T86597 C5ADP4 56950567 IC50 = 9000 nM T86597 CFW0D1 57339435 IC50 = 794.33 nM T86597 CF8B4E 60498769 IC50 = 59000 nM T86597 CPY59D 67195867 IC50 = 50118.72 nM T86597 CN3KZ8 68161075 IC50 = 501.19 nM T86597 C49IOA 68161669 IC50 = 794.33 nM T86597 CJ7N3M 68184870 IC50 = 1258.93 nM T86597 CT4Z2A 68184871 IC50 = 630.96 nM T86597 CEX74I 68186034 IC50 = 10000 nM T86597 C25INY 68204735 IC50 = 2511.89 nM T86597 CMC7V5 70664240 IC50 = 1995.26 nM T86597 C1I6OH 70681167 IC50 = 12589.25 nM T86597 C7GJW9 70681170 IC50 = 501.19 nM T86597 C8H4JX 70681173 IC50 = 1000 nM T86597 C6NYK2 70681174 IC50 = 501.19 nM T86597 C8KBJ0 70683271 IC50 = 1995.26 nM T86597 CXD3F9 70691699 IC50 = 501.19 nM T86597 CL8Y9N 71450297 IC50 = 1584.89 nM T86597 C6CQT5 71462842 IC50 = 3162.28 nM T86597 CIPN50 71760902 Ki = 14 nM T86597 C2AFW1 72702849 IC50 = 1258.93 nM T86597 C3R1IL 72703043 IC50 = 100000 nM T86597 CK9O6W 72705811 IC50 = 31622.78 nM T86597 C5TB9S 77843982 Ki = 27 nM T86597 CS6XE0 77846025 Ki = 11.1 nM T86597 COZ8S1 78319129 Ki = 160 nM T86597 C4IF8T 78425807 Ki = 0.48 nM T86597 CFE7R3 86270928 Ki = 2.5 nM T86597 C53QEW 86669224 IC50 = 15848.93 nM T86597 CEDL57 89657555 IC50 = 16 nM T86597 CZJ8W9 90387575 Ki = 15.4 nM T86597 CU91GC 105539824 IC50 = 20000 nM T86597 C1W3XP 112499930 IC50 = 1600 nM T86597 CYX7T2 117072549 IC50 > 100000 nM T86597 CPN74M 118719856 IC50 = 794.33 nM T86597 CE8DL3 118719857 IC50 = 1000 nM T86597 COEU47 118719858 IC50 = 1995.26 nM T86597 CX05SW 118719859 IC50 = 1258.93 nM T86597 CRCG07 118719860 IC50 = 794.33 nM T86597 C03XDG 118719861 IC50 = 794.33 nM T86597 C3ML2F 118719862 IC50 = 1258.93 nM T86597 CZ67WF 118719863 IC50 = 25118.86 nM T86597 C0HR9Y 118719864 IC50 = 501.19 nM T86597 C7F4EP 118719865 IC50 = 1000 nM T86597 CA40QV 118719866 IC50 = 1258.93 nM T86597 CZ8QI6 118719867 IC50 = 1584.89 nM T86597 C8NRI9 118719868 IC50 = 1258.93 nM T86597 C3Y2WT 118719869 IC50 = 1584.89 nM T86597 C52HPM 118719870 IC50 = 630.96 nM T86597 CUT97H 118719871 IC50 = 630.96 nM T86597 CBE68N 118719872 IC50 = 1000 nM T86597 C29WRE 118719873 IC50 = 794.33 nM T86597 C8J0TY 118719874 IC50 = 1995.26 nM T86597 CZR10C 118719875 IC50 = 3981.07 nM T86597 C35AWU 118719876 IC50 = 6309.57 nM T86597 C87ZPY 118796358 IC50 > 100000 nM T86597 C9MQF0 119098887 IC50 = 33234 nM T86597 C0QX4D 119098889 IC50 = 50857 nM T86597 C4ITM8 122180892 IC50 = 23000 nM T86597 CFCA87 122180893 IC50 = 24000 nM T86597 CZRJ29 122180894 IC50 = 13000 nM T86597 C8RE2M 122180895 IC50 > 50000 nM T86597 C54NBV 122180896 IC50 = 13000 nM T86597 C26RAL 122180897 IC50 = 26000 nM T86597 CC35RW 122180898 IC50 = 5000 nM T86597 C7E3VM 122180899 IC50 = 25000 nM T86597 C2UQW0 122180900 IC50 > 50000 nM T86597 C67LPS 122180901 IC50 = 10000 nM T86597 C3FC0Z 122180902 IC50 = 12000 nM T86597 CSR48T 122180903 IC50 = 49000 nM T86597 CVI96R 122180904 IC50 > 50000 nM T86597 CXP8T3 122180909 IC50 = 12000 nM T86597 C3QJ5L 122181550 IC50 > 31622.78 nM T86597 CLI1P6 122235215 EC50 = 480 nM T86597 C4GYP3 126521168 IC50 = 43 nM T86597 CL2PG5 126521180 IC50 = 52 nM T86597 CQV90I 126521354 IC50 = 185 nM T86597 C0HJV7 126521430 IC50 > 999 nM T86597 CN6FI1 126521537 IC50 = 6 nM T86597 C1DOG4 126521586 IC50 = 25 nM T86597 CRY0S6 126563516 IC50 = 38 nM T86597 CN0D6M 126563562 IC50 = 34 nM T86597 CKB36S 126563576 IC50 = 25 nM T86597 CX79NH 126563597 IC50 = 44 nM T86597 C2K5XG 126563611 IC50 = 95 nM T86597 CZ06NR 126563612 IC50 = 45 nM T86597 CM5P2Z 126563615 IC50 = 40 nM T86597 C15ILF 126564427 IC50 = 28 nM T86597 CROY39 126564463 IC50 = 25 nM T86597 CHO12Y 126564469 IC50 > 10000 nM T86597 CB2AS4 126564470 IC50 = 33 nM T86597 CBW08I 126564471 IC50 = 39 nM T86597 CD78GB 126564481 IC50 = 25 nM T86597 CU8CA9 126564486 IC50 = 17 nM T86597 CQW6P1 126564822 IC50 = 24 nM T86597 CQS5T2 126564831 IC50 = 204 nM T86597 CNP2L7 126564832 IC50 = 18 nM T86597 C58PNK 126564833 IC50 = 37 nM T86597 CHPV09 126564847 IC50 = 3 nM T86597 CJZW04 126564858 IC50 = 20 nM T86597 CH14FC 127032939 IC50 = 6600 nM T86597 CS4NG8 127033568 IC50 = 30000 nM T86597 CGA71L 127048256 IC50 = 59555 nM T86597 CH6T5J 127048257 IC50 = 30330 nM T86597 C60SZQ 127048258 IC50 = 21687 nM T86597 C50BMV 127049279 IC50 = 5876 nM T86597 CTF4N2 127051087 IC50 > 100000 nM T86597 CLSZ47 127051725 IC50 = 16654 nM T86597 CMY93U 127051726 IC50 > 100000 nM T86597 CY8V1A 127051727 IC50 > 100000 nM T86597 CXZT48 127052023 IC50 > 100000 nM T86597 C9L1OG 130345579 Ki = 1.7 nM T86597 CTDG89 135141500 IC50 = 830 nM T86597 CF2BU6 135141501 IC50 = 410 nM T86597 CBC37Z 135141502 IC50 = 1910 nM T86597 C12HJT 135141503 IC50 = 1400 nM T86597 C50NEZ 135141504 IC50 = 1080 nM T86597 CRNY32 135397673 Ki = 0.27 nM T86597 C5F3LV 135567026 IC50 = 24600 nM T86597 CO71RI 137285009 IC50 = 1836 nM T86597 CS9MR6 137285011 IC50 = 803 nM T86597 CFXE14 137321203 IC50 = 100 nM T86597 CXN4U1 137321204 IC50 = 316.23 nM T86597 C4VNB8 137369426 IC50 = 147 nM T86597 CU5N8O 137701509 IC50 = 29000 nM T86597 CQ6XB7 139030526 IC50 = 19952.62 nM T86597 C1G9LA 139035062 Ki = 3.1 nM T86597 CG6X3A 142535938 IC50 = 35 nM T86597 CD6U7X 145925666 IC50 = 8948 nM T86597 C1HLK5 145951928 IC50 = 44 nM T86597 CV83ED 145972103 Ki = 2.6 nM T86597 CK20BY 145988169 Ki = 57.3 nM T86597 C9FIY4 153534005 IC50 = 16400 nM T86597 CFD6H1 155352361 IC50 = 30000 nM T86597 CFK2B1 155352401 IC50 > 250000 nM T86597 C76QMK 155513141 Ki = 8.9 nM T86597 C27LFN 155514936 IC50 = 1800 nM T86597 C6OP0S 155535292 Ki = 9.1 nM T86597 C0HI7N 155536879 IC50 = 997 nM T86597 CUX25H 155547195 Ki = 19.1 nM T86597 CZA5N1 155561689 IC50 > 45000 nM T86597 C7ICA9 155564455 IC50 = 78 nM T86597 D00XRH 91820725 IC50 = 3981.07 nM T86597 D03LIP 13953710 IC50 = 29.9 nM T86597 D09VHS 3971 IC50 = 7400 nM T86597 D0F5TZ 91827383 IC50 = 6309.57 nM T86597 D0H3TC 54669868 IC50 = 1600 nM T86597 D0T3AT 672548 IC50 = 28000 nM T86597 D0WU1S 52912189 Ki = 9 nM T69685 D0M8AB 750 IC50 = 31600 nM T69685 D05WWJ 6604909 IC50 = 0.39 nM T69685 D0LT0U 11717074 IC50 = 100 nM T69685 D0O0BM 44156901 Ki = 11.6 nM T69685 D0R8HY 15951941 IC50 = 29 nM T69685 D06SBS 9954540 IC50 = 80.1 nM T69685 D0U1HP 23670635 IC50 = 316.23 nM T69685 CBGO28 70419 EC50 > 10000 nM T69685 C16UJV 2916853 EC50 = 1300 nM T69685 CCO5Y6 4092325 EC50 > 10000 nM T69685 C7B2UD 4154232 IC50 > 200000 nM T69685 CL5BU6 4639181 IC50 > 200000 nM T69685 C4PJ1X 5311286 IC50 > 100 nM T69685 CUY2A3 5311287 IC50 > 100 nM T69685 C3TR2C 6436908 IC50 > 30000 nM T69685 CK1OS6 6437024 IC50 > 3000 nM T69685 CCH5V1 6913738 IC50 > 10000 nM T69685 C8Z6VJ 9225008 EC50 > 10000 nM T69685 C2LBO0 9800357 IC50 = 580 nM T69685 CJP84L 9802774 IC50 = 130 nM T69685 C5L6CA 9828521 IC50 = 155 nM T69685 CF2P5Q 9925334 IC50 = 590 nM T69685 C38YCX 10126825 IC50 = 150 nM T69685 C45HMS 10172780 IC50 = 160 nM T69685 CE6Q4F 10193969 IC50 = 1000 nM T69685 CECW60 10194073 IC50 = 53000 nM T69685 CUN2W9 10215851 IC50 = 1258.93 nM T69685 C6S8WQ 10236952 IC50 = 12589.25 nM T69685 CRC3A1 10237135 IC50 = 7943.28 nM T69685 CR1CA4 10286974 IC50 = 794.33 nM T69685 CD2K6P 10308908 IC50 = 3162.28 nM T69685 CZS7V2 10915847 IC50 > 100 nM T69685 CKL5O9 11059011 IC50 > 100 nM T69685 CV91EB 11153218 EC50 = 6287 nM T69685 C76YFB 11155030 EC50 = 70 nM T69685 CFO4R6 11155673 IC50 = 5.7 nM T69685 CH72UP 11156047 EC50 = 15 nM T69685 CSQA43 11188596 EC50 = 682 nM T69685 CUBX19 11189444 EC50 = 56 nM T69685 C49LGB 11190646 EC50 = 4563 nM T69685 COQF79 11198976 EC50 > 30000 nM T69685 C4EUH1 11202082 EC50 = 20 nM T69685 C4SP5J 11202309 EC50 = 433 nM T69685 CUV92K 11211923 EC50 = 48 nM T69685 CS5ET8 11212373 EC50 = 70 nM T69685 C54NSQ 11214321 EC50 = 29 nM T69685 C73SKC 11223162 EC50 = 15237 nM T69685 C26MVG 11223982 EC50 = 450 nM T69685 CO79MA 11225426 EC50 = 40 nM T69685 CWX3G9 11225589 EC50 = 16728 nM T69685 C2EY1P 11237095 EC50 = 8 nM T69685 C9EW5N 11245541 EC50 = 979 nM T69685 CX43IH 11248146 EC50 = 10 nM T69685 CQD4L6 11248803 EC50 = 31 nM T69685 CP0C2Q 11257803 EC50 = 1419 nM T69685 CVP4L6 11269915 EC50 = 281 nM T69685 CP28LW 11282509 EC50 = 73 nM T69685 CQR3W4 11283425 EC50 = 33 nM T69685 C76QCL 11293598 EC50 = 77 nM T69685 CXL1I8 11294866 EC50 = 25 nM T69685 CVH5B3 11317032 EC50 = 1212 nM T69685 C8S4FU 11317045 EC50 = 16 nM T69685 C61LSX 11325613 IC50 = 3900 nM T69685 CTG7D3 11326273 IC50 = 9200 nM T69685 CQ0H8E 11328142 EC50 = 69 nM T69685 CP3S5J 11337188 EC50 = 970 nM T69685 CS1W7V 11338717 EC50 = 423 nM T69685 C0J6KU 11349288 EC50 = 787 nM T69685 CX02EN 11363500 EC50 = 91 nM T69685 C7I4FX 11363702 IC50 = 2.4 nM T69685 CCAX86 11372350 IC50 = 380 nM T69685 CQC4G5 11372671 EC50 = 77 nM T69685 C3EU2G 11373827 EC50 > 30000 nM T69685 CV71EO 11396919 EC50 = 15 nM T69685 C3NWX6 11405950 IC50 = 70 nM T69685 CGO58L 11406629 EC50 = 4 nM T69685 CBJ0X5 11407510 EC50 = 350 nM T69685 CD90BT 11417036 EC50 = 1466 nM T69685 CW0E4L 11418847 EC50 = 393 nM T69685 CCF0L6 11429237 EC50 = 525 nM T69685 CO0Y4L 11429888 EC50 = 16000 nM T69685 CHQ3N0 11439977 IC50 = 7300 nM T69685 CJG2M6 11441323 EC50 = 99 nM T69685 CZO4Q8 11441561 EC50 = 73 nM T69685 C5P4KW 11452904 EC50 = 419 nM T69685 C6BK7A 11454048 IC50 = 2.6 nM T69685 CA2R1I 11462855 EC50 > 30000 nM T69685 CKIQ83 11463791 EC50 = 284 nM T69685 CY3AK9 11464241 EC50 = 5610 nM T69685 CC9TX5 11464294 EC50 = 563 nM T69685 CP0AY1 11465204 EC50 = 1 nM T69685 CRU3C9 11465585 EC50 = 12 nM T69685 CAY3P0 11488045 EC50 = 39 nM T69685 CHT5Y8 11488238 EC50 = 12 nM T69685 C9N7BP 11488921 EC50 = 47 nM T69685 CYFU19 11496738 IC50 = 2.5 nM T69685 CHV9P4 11503316 IC50 = 3 nM T69685 CWNS78 11503732 IC50 = 6.6 nM T69685 C8K6LT 11503999 IC50 = 3 nM T69685 CGWZ71 11510618 IC50 = 30 nM T69685 C0P9VC 11517722 IC50 = 11.9 nM T69685 CMEK74 11518581 EC50 = 15 nM T69685 C4OAQ8 11518805 EC50 = 17 nM T69685 CHGW75 11539784 IC50 = 57 nM T69685 CW2IZ4 11540267 EC50 = 21 nM T69685 C2JQ1P 11569401 EC50 = 13 nM T69685 C9CT2I 11583046 IC50 = 300 nM T69685 CAR70B 11583581 IC50 = 200 nM T69685 CELV43 11597407 EC50 = 30 nM T69685 C15TEH 11604449 IC50 = 26 nM T69685 C4NMD3 11619325 IC50 = 6.9 nM T69685 C41ASM 11620014 IC50 = 3.5 nM T69685 CCB89R 11620302 IC50 = 2 nM T69685 C6SPR0 11627103 EC50 = 16 nM T69685 CWA91I 11641652 IC50 = 4.33 nM T69685 CIJ40B 11641798 EC50 = 14 nM T69685 CJ6PI1 11647944 EC50 = 28 nM T69685 C8R4DN 11656017 IC50 = 10.35 nM T69685 CHBN05 11662843 IC50 = 9.7 nM T69685 CKI68D 11663033 EC50 = 30 nM T69685 CW9H0I 11677151 IC50 = 4.4 nM T69685 C01ORH 11691531 EC50 = 50 nM T69685 CWK01R 11699068 IC50 = 2.4 nM T69685 CD91SM 11699654 IC50 = 412 nM T69685 CN4WC9 11705483 IC50 = 220 nM T69685 CV3P7H 11712529 IC50 = 77 nM T69685 CHJ0F2 11739625 IC50 = 7800 nM T69685 CV8CF3 11749578 EC50 = 232 nM T69685 CPYN49 11772006 IC50 = 5100 nM T69685 CY04HA 11854550 EC50 = 57 nM T69685 C8P9GD 11966041 IC50 = 1.89 nM T69685 C4I3RS 12307852 IC50 > 200000 nM T69685 CQ1CJ6 14013470 IC50 = 549 nM T69685 CSLB93 15951662 IC50 = 3333 nM T69685 C1TCV5 15951943 IC50 = 36.9 nM T69685 CHPY30 15952325 IC50 = 132.4 nM T69685 CD7K0Y 15965865 EC50 = 26 nM T69685 C7Q8IN 15984044 IC50 = 59 nM T69685 CDR71P 16043240 EC50 = 61 nM T69685 CERP08 16219807 IC50 = 125.89 nM T69685 CG3CF0 16678871 IC50 = 9.5 nM T69685 C5U7JX 16678872 IC50 = 21.2 nM T69685 C4YMP1 16725956 Ki = 15.9 nM T69685 C2L9HN 16960944 EC50 = 32000 nM T69685 C9EAP4 18098131 EC50 = 500 nM T69685 C87WIK 18104758 EC50 = 110 nM T69685 C5Q4FX 18441731 EC50 = 24 nM T69685 C8AZW7 18441735 EC50 = 44 nM T69685 C1Y8DF 21082542 EC50 = 1953 nM T69685 C0BMI8 21082546 EC50 = 1394 nM T69685 CA24YC 21082547 EC50 = 127 nM T69685 CO48CY 21082549 EC50 = 18646 nM T69685 C4GL6C 21082550 EC50 = 158 nM T69685 CB8CM1 21082551 EC50 = 1313 nM T69685 CU14BE 21082552 EC50 = 2638 nM T69685 C1D2AZ 21082553 EC50 = 69 nM T69685 C6UXT7 21082554 EC50 = 132 nM T69685 CME6O3 21082560 EC50 = 127 nM T69685 CUG70N 21082561 EC50 > 30000 nM T69685 C2SRF0 21082562 EC50 > 30000 nM T69685 C4VW7M 21082563 EC50 = 4480 nM T69685 CCKW02 21082574 EC50 = 270 nM T69685 C84XQE 21082576 EC50 = 1131 nM T69685 C9XQS4 21082577 EC50 = 113 nM T69685 CJ7IZ4 22046253 IC50 = 290 nM T69685 CE65DB 22115679 Ki = 500 nM T69685 CS7E2L 24532923 EC50 = 1900 nM T69685 CZ03FI 24649020 EC50 = 1100 nM T69685 CQ35ZB 24743795 EC50 = 16 nM T69685 CYM02E 24847114 EC50 = 72 nM T69685 CDI7N3 24897002 EC50 = 89 nM T69685 C8GN9W 24899993 EC50 = 88 nM T69685 CZSA05 24899995 EC50 = 25 nM T69685 CIZ6O1 24900235 EC50 = 33 nM T69685 C61ARF 24900236 EC50 = 56 nM T69685 CGO5X4 24946690 Ki = 47 nM T69685 C7UD6F 24957934 IC50 = 45 nM T69685 C8AL2P 25207063 IC50 = 41 nM T69685 C8U4KM 26365758 EC50 = 700 nM T69685 CR8IG7 29297108 EC50 = 400 nM T69685 CO74NY 41772744 EC50 = 120 nM T69685 CPF50A 44184875 EC50 = 30 nM T69685 C8ARJ4 44190514 IC50 > 3000 nM T69685 C8GUW6 44303464 IC50 = 501.19 nM T69685 CM2H7W 44303471 IC50 = 31622.78 nM T69685 CCF58H 44303473 IC50 = 398.11 nM T69685 C7NT1B 44303490 IC50 = 5011.87 nM T69685 C6WCG8 44303494 IC50 = 1258.93 nM T69685 CS17HT 44303504 IC50 = 251.19 nM T69685 CT30FL 44303505 IC50 = 100 nM T69685 CH92YI 44303507 IC50 = 2511.89 nM T69685 CRT3I7 44303531 IC50 = 12589.25 nM T69685 C6CXZ2 44303544 IC50 = 19952.62 nM T69685 C8VBE6 44303548 IC50 = 100000 nM T69685 CCY0S6 44303558 IC50 = 2511.89 nM T69685 C0RM8L 44303561 IC50 = 11748.98 nM T69685 CU1S2F 44303570 IC50 = 3981.07 nM T69685 C7K5OC 44303575 IC50 = 977.24 nM T69685 CXG7Q1 44303577 IC50 = 2630.27 nM T69685 CX5QC4 44303583 IC50 = 501.19 nM T69685 C45QRK 44303607 IC50 = 446.68 nM T69685 CZ12JO 44303616 IC50 = 151.36 nM T69685 CMPG81 44303910 IC50 = 1000 nM T69685 CRN2F0 44303927 IC50 = 100000 nM T69685 C4M2XD 44392941 IC50 > 50000 nM T69685 CK8M2N 44392949 IC50 = 18000 nM T69685 CG1Y7S 44392954 IC50 = 1500 nM T69685 CJR60W 44392970 IC50 = 16000 nM T69685 CR67NU 44392971 IC50 > 10000 nM T69685 C6O7EV 44392976 IC50 = 1600 nM T69685 CH62JZ 44392977 IC50 = 4600 nM T69685 C79IFE 44392991 IC50 = 1700 nM T69685 C8F1PT 44392992 IC50 > 10000 nM T69685 CQV96A 44393002 IC50 = 550 nM T69685 CA54ME 44393005 IC50 = 360 nM T69685 C47NYM 44393006 IC50 = 3600 nM T69685 C5VWI4 44393009 IC50 = 22000 nM T69685 C1NDZ3 44393014 IC50 = 1700 nM T69685 C1BZC2 44393024 IC50 = 1900 nM T69685 CXO6R9 44393035 IC50 = 1400 nM T69685 CB7F1Q 44393038 IC50 = 2900 nM T69685 C1A6KR 44393043 IC50 > 1000 nM T69685 CW9QG2 44406457 EC50 = 140 nM T69685 CGN73V 44406458 EC50 = 62 nM T69685 CJ2K3A 44406465 EC50 = 9000 nM T69685 C9X2ED 44406466 EC50 = 17000 nM T69685 CQ4AS2 44406469 EC50 = 4400 nM T69685 C0J7IK 44406489 EC50 = 26 nM T69685 C5TIM4 44406497 EC50 = 80 nM T69685 C7EIC2 44406499 EC50 = 29000 nM T69685 C5SQ1C 44406502 EC50 > 3000 nM T69685 CBUR32 44406503 EC50 = 24 nM T69685 C17FYG 44406538 EC50 = 44 nM T69685 C07CNE 44406539 EC50 = 261 nM T69685 C5DGV2 44406540 EC50 = 130 nM T69685 C9Z0ET 44406541 EC50 = 15 nM T69685 C1L8CG 44406543 EC50 = 24 nM T69685 CP1OZ6 44406544 EC50 = 99 nM T69685 CR5WZ2 44406546 EC50 = 1500 nM T69685 CS04TK 44406550 EC50 = 130 nM T69685 C8HRC9 44406551 EC50 = 130 nM T69685 C8XHL1 44406552 EC50 = 65 nM T69685 C21FWX 44406553 EC50 = 66 nM T69685 CSPE30 44406557 EC50 = 110 nM T69685 C1LVU2 44406558 EC50 = 450 nM T69685 CPG5O7 44406559 EC50 = 55 nM T69685 CCV3E6 44406563 EC50 = 400 nM T69685 CEI1H6 44406577 EC50 = 630 nM T69685 C09APK 44406579 EC50 > 30000 nM T69685 CH4QB6 44406580 EC50 = 6600 nM T69685 CD7Y0Z 44406585 EC50 = 34 nM T69685 CC15BY 44406587 EC50 = 173 nM T69685 C2MV0K 44406589 EC50 = 49 nM T69685 C7VYD6 44406590 EC50 = 3300 nM T69685 C1IM9R 44406603 EC50 = 40 nM T69685 C3VE8N 44406604 EC50 = 50 nM T69685 C2JG5K 44406608 EC50 = 25 nM T69685 CCI5Z1 44406618 EC50 = 73 nM T69685 C7ES2W 44406621 EC50 = 56 nM T69685 C0MX1J 44406626 EC50 = 258 nM T69685 C0SKT9 44406641 EC50 = 25 nM T69685 CHF65L 44406659 EC50 = 510 nM T69685 CUAZ73 44406660 EC50 = 6600 nM T69685 C9PK5G 44406666 EC50 = 1100 nM T69685 CP91RV 44406667 EC50 = 1700 nM T69685 CZNQ19 44406672 EC50 = 24 nM T69685 CL58DU 44406677 EC50 = 5300 nM T69685 C38ABN 44406682 EC50 = 58 nM T69685 CZ65PF 44406685 EC50 = 90 nM T69685 COHV70 44406692 EC50 = 750 nM T69685 CMR3C6 44406693 EC50 = 65 nM T69685 C79LAD 44406694 EC50 = 7400 nM T69685 CTK1J4 44406698 EC50 = 7300 nM T69685 CIR94D 44406707 EC50 = 23 nM T69685 CC1A9V 44406708 EC50 = 40 nM T69685 CB36AF 44406709 EC50 = 85 nM T69685 C4M1GV 44406714 EC50 = 610 nM T69685 CKW8U6 44406718 EC50 = 9300 nM T69685 CWY76P 44406719 EC50 = 27 nM T69685 CC6SW1 44406725 EC50 = 130 nM T69685 CYA4I3 44406726 EC50 = 67 nM T69685 C75ZOH 44406728 EC50 = 1800 nM T69685 C8P6KZ 44408650 IC50 = 1200 nM T69685 CD02UB 44408668 IC50 = 6.4 nM T69685 COE9P8 44408677 IC50 = 19 nM T69685 C9A3KX 44408684 IC50 = 1300 nM T69685 C26OCQ 44408698 IC50 = 0.47 nM T69685 CU9N6P 44408780 IC50 = 2800 nM T69685 C79THI 44408783 IC50 = 103 nM T69685 CHLZ29 44408889 IC50 = 2.9 nM T69685 CGO43S 44408913 IC50 = 1.9 nM T69685 C63NOZ 44408919 IC50 = 0.95 nM T69685 CB1X5Y 44408943 IC50 = 28 nM T69685 CX4LY5 44408947 IC50 = 19 nM T69685 C1XOH2 44408964 IC50 = 85 nM T69685 CK4VS3 44414119 IC50 = 160 nM T69685 CMOX45 44414308 IC50 > 50000 nM T69685 C6G3UW 44414326 IC50 = 11000 nM T69685 CB1GM9 44414328 IC50 = 160 nM T69685 CUV6A9 44414329 IC50 = 300 nM T69685 CO67RG 44414358 IC50 = 1400 nM T69685 CHE9U0 44414452 IC50 = 600 nM T69685 C9JCE4 44414453 IC50 = 19000 nM T69685 CBFN50 44414478 IC50 = 1200 nM T69685 CH0PL8 44414479 IC50 = 400 nM T69685 C8Q6EH 44414494 IC50 = 950 nM T69685 C65REV 44414517 IC50 = 520 nM T69685 CNRM76 44414568 IC50 = 18000 nM T69685 CJ4BR0 44414569 IC50 = 12000 nM T69685 C4EOX7 44414587 IC50 = 8900 nM T69685 CZR7N0 44414588 IC50 = 26000 nM T69685 CD0SY5 44414617 IC50 = 50000 nM T69685 CE7KR2 44414618 IC50 = 22000 nM T69685 CPG8E9 44414638 IC50 = 30000 nM T69685 CK7NA6 44414639 IC50 = 15000 nM T69685 CZ04TL 44414640 IC50 = 47000 nM T69685 CC2M5E 44414664 EC50 = 147 nM T69685 C3J4VM 44414717 EC50 = 62 nM T69685 CXC04Z 44414729 EC50 = 2830 nM T69685 C6O2VL 44414730 EC50 = 246 nM T69685 C7N9AR 44414747 EC50 = 2880 nM T69685 C1BKH2 44414770 EC50 = 474 nM T69685 CY49WT 44414777 EC50 = 139 nM T69685 CP63GQ 44414781 EC50 > 30000 nM T69685 CRCQ06 44414830 EC50 = 1064 nM T69685 C1PK7O 44414844 EC50 = 1296 nM T69685 C5Z9VE 44414845 EC50 = 36 nM T69685 C4LI9Q 44414865 EC50 = 43 nM T69685 CWR4S6 44414876 EC50 = 93 nM T69685 CU5WF7 44414888 EC50 = 229 nM T69685 CEN9K5 44414889 EC50 = 113 nM T69685 CDEC-35 44420018 IC50 = 181 nM T69685 CLJ58G 44420020 IC50 = 517 nM T69685 CJP9Y2 44420021 IC50 = 544 nM T69685 CZ54MW 44420030 IC50 = 472 nM T69685 C69SHV 44420039 IC50 = 264 nM T69685 CVL2E6 44420041 IC50 > 5000 nM T69685 CQ43MW 44420042 IC50 = 88.4 nM T69685 C2ETD8 44420043 IC50 = 12.6 nM T69685 C65CVW 44420046 IC50 = 69 nM T69685 C5K7BH 44420047 IC50 = 109 nM T69685 CE20MW 44420048 IC50 = 42.8 nM T69685 CLWG78 44420049 IC50 = 67.8 nM T69685 CCB3V7 44420052 IC50 > 5000 nM T69685 CW90RA 44420055 IC50 > 5000 nM T69685 CHAE84 44420063 IC50 > 5000 nM T69685 CY4B7E 44420069 IC50 > 5000 nM T69685 CWKV41 44420132 IC50 = 8.4 nM T69685 C8AZ0R 44420133 IC50 = 12.5 nM T69685 C8ILS1 44420139 IC50 = 6.3 nM T69685 C7H0UM 44420140 IC50 = 131 nM T69685 CP2YG8 44423663 IC50 > 30000 nM T69685 CY9IK3 44438461 Ki = 394 nM T69685 C6W2EZ 44438462 Ki = 134 nM T69685 C9IFR5 44438464 Ki = 26.8 nM T69685 CUB30F 44438465 Ki = 66.8 nM T69685 CE36YV 44438467 Ki = 61.4 nM T69685 CLWE65 44438469 Ki = 108 nM T69685 CI93VE 44438472 Ki = 10.2 nM T69685 CXD9B1 44438473 Ki = 11 nM T69685 C0QEB9 44438474 Ki = 85.3 nM T69685 CJ48AY 44439739 IC50 = 1000 nM T69685 CZL04F 44439740 IC50 = 1000 nM T69685 CQ1WX7 44439741 IC50 = 199.53 nM T69685 CH6LN5 44439742 IC50 = 501.19 nM T69685 C0QAK9 44439762 IC50 = 1584.89 nM T69685 CY3A4E 44439768 IC50 = 3162.28 nM T69685 CPT6U1 44439769 IC50 = 2511.89 nM T69685 CG86RM 44439770 IC50 = 6309.57 nM T69685 CE6HL3 44439789 IC50 = 316.23 nM T69685 CR0WT3 44439790 IC50 = 7943.28 nM T69685 C9S7IU 44439791 IC50 = 100 nM T69685 CFU7G5 44439792 IC50 = 3981.07 nM T69685 CP4HU2 44439793 IC50 = 3981.07 nM T69685 CFG10D 44439794 IC50 = 1000 nM T69685 CI27KN 44439796 IC50 = 3981.07 nM T69685 CO75SU 44439798 IC50 = 2511.89 nM T69685 C0Z9NW 44439800 IC50 = 3162.28 nM T69685 CF0A3Z 44439801 IC50 = 3162.28 nM T69685 CC0MF2 44439803 IC50 = 3162.28 nM T69685 C8MJX3 44444240 IC50 = 175 nM T69685 CY1M5B 44444241 IC50 = 26 nM T69685 CJ4MN5 44444243 IC50 = 68 nM T69685 C2PD4R 44444244 IC50 = 632 nM T69685 C1DG6B 44444245 IC50 = 45 nM T69685 CP20CO 44444246 IC50 = 59 nM T69685 CSK28U 44444247 IC50 = 104 nM T69685 C3QTF8 44444248 IC50 = 27 nM T69685 CM08FN 44444249 IC50 = 18 nM T69685 C39BVE 44444250 IC50 = 76 nM T69685 CA1YH0 44444251 IC50 = 834 nM T69685 C6EQ9M 44444254 IC50 = 19 nM T69685 CB6Q4T 44444255 IC50 = 702 nM T69685 CXEP90 44444258 IC50 = 40 nM T69685 CUI25H 44444260 IC50 = 65 nM T69685 C0R3PZ 44444261 IC50 = 85 nM T69685 C1W5TQ 44444262 IC50 = 229 nM T69685 CT9O7J 44444263 IC50 = 70 nM T69685 C1QIO5 44444264 IC50 = 289 nM T69685 C9NDY4 44444265 IC50 = 251 nM T69685 CRI72W 44444267 IC50 = 53 nM T69685 CS9R1C 44444268 IC50 = 674 nM T69685 CUF89R 44444270 IC50 = 965 nM T69685 CA1O3V 44444271 IC50 = 108 nM T69685 CJSA47 44444273 IC50 = 56 nM T69685 CHUJ64 44444275 IC50 = 351 nM T69685 CCMV69 44444276 IC50 = 139 nM T69685 C4X3EO 44444281 IC50 = 957 nM T69685 CX46JK 44444284 IC50 = 496 nM T69685 C7QHD4 44444287 IC50 = 161 nM T69685 C29RVP 44444289 IC50 = 28 nM T69685 CI0D3P 44444290 IC50 = 34 nM T69685 CI1T0P 44444291 IC50 = 12 nM T69685 C3Y5MT 44444292 IC50 = 25 nM T69685 CUAK74 44444294 IC50 = 14 nM T69685 CX47CG 44444296 IC50 = 17 nM T69685 C2GF7J 44444298 IC50 = 13 nM T69685 CYQX20 44465025 Ki = 3 nM T69685 C5D9US 44564632 IC50 = 2592 nM T69685 C0VP3T 44564633 IC50 = 661 nM T69685 CSX63M 44564634 IC50 = 576 nM T69685 CA87MB 44564635 IC50 = 17.7 nM T69685 CDC0B2 44564672 IC50 = 4 nM T69685 CY5W2O 44564673 IC50 = 69.3 nM T69685 C8F9IZ 44564674 IC50 = 79.3 nM T69685 CF2TP7 44564679 IC50 = 2.9 nM T69685 CTJ49O 44564680 IC50 = 26.5 nM T69685 CCL8B7 44564681 IC50 = 2.8 nM T69685 C1TRY8 44564708 IC50 = 3314 nM T69685 C93RCB 44564709 IC50 = 148 nM T69685 CBOT51 44564710 IC50 = 58.9 nM T69685 C9M2AU 44564718 IC50 = 17.7 nM T69685 C1TB6K 44564719 IC50 = 38.1 nM T69685 C4E8MC 44564755 IC50 = 43.1 nM T69685 C23BWM 44564765 IC50 = 86 nM T69685 CQN60Y 44564766 IC50 = 9.7 nM T69685 C6U8ZL 44564801 IC50 = 120 nM T69685 C3FB7K 44564831 IC50 > 5000 nM T69685 C7HKG5 44564832 IC50 = 1070 nM T69685 C5VIN0 44565248 IC50 = 107 nM T69685 COR7F4 44565249 IC50 = 49.4 nM T69685 CS2I4V 44565250 IC50 = 19.5 nM T69685 C7FE5L 44565251 IC50 = 129 nM T69685 C20DZB 44565252 IC50 = 48.3 nM T69685 C7URY2 44565253 IC50 = 6.9 nM T69685 CQV4K2 44565260 IC50 = 833 nM T69685 CG21WE 44565261 IC50 = 31.3 nM T69685 C4PAC2 44565262 IC50 = 19.4 nM T69685 C2XJY7 44565263 IC50 = 38.3 nM T69685 CH4GW0 44565264 IC50 = 54.7 nM T69685 C8I3SF 44565265 IC50 = 7.4 nM T69685 C9UO1Z 44565266 IC50 > 5000 nM T69685 CW1J3T 44565267 IC50 = 482 nM T69685 C7WL4C 44565270 IC50 = 103 nM T69685 CC1O6M 44565271 IC50 = 517 nM T69685 C6EAC3 44565272 IC50 = 131 nM T69685 C5LN0C 44578913 IC50 = 154 nM T69685 CG80OC 44578914 EC50 = 4790 nM T69685 C7LAT0 44578954 EC50 = 1800 nM T69685 CBG04P 44578955 EC50 = 390 nM T69685 CA3FO8 44578956 EC50 = 230 nM T69685 CA16QJ 44578957 EC50 = 6630 nM T69685 CFH01N 44578958 EC50 = 4100 nM T69685 CMA26F 44578959 EC50 = 730 nM T69685 C79PYS 44578960 EC50 = 1270 nM T69685 CF39ON 44578961 EC50 > 10000 nM T69685 C4KI0B 44579189 EC50 = 200 nM T69685 C1I0QG 44579190 EC50 > 10000 nM T69685 C6VFZ3 44579191 EC50 > 10000 nM T69685 C1O5ET 44579232 EC50 = 4050 nM T69685 CY8NJ4 44579233 EC50 = 300 nM T69685 CSLC36 44579234 EC50 = 5050 nM T69685 CBK23W 44579235 EC50 > 10000 nM T69685 CS2KV6 44579236 EC50 > 10000 nM T69685 C60CAD 44579237 EC50 > 10000 nM T69685 CX85MD 44579273 EC50 > 10000 nM T69685 CO7MU4 44580053 EC50 = 16 nM T69685 CY7MA0 44580054 EC50 > 10000 nM T69685 CI24ZU 44580055 EC50 = 1400 nM T69685 C86GWQ 44580106 EC50 = 7100 nM T69685 CF5ST4 44580229 EC50 = 530 nM T69685 CH1G5K 44580230 EC50 = 1100 nM T69685 CBLJ49 44580260 EC50 = 2900 nM T69685 C1UO6X 44580261 EC50 = 310 nM T69685 C1FNB8 44580262 EC50 = 100 nM T69685 CYA4U0 44580302 EC50 = 78 nM T69685 C4EK3O 44580303 EC50 = 110 nM T69685 COY93Q 44580304 EC50 = 30 nM T69685 CX16RS 44580305 EC50 = 40 nM T69685 CD9M8A 44580340 EC50 = 41 nM T69685 CT5FH1 44580341 EC50 = 37 nM T69685 CE86ZK 44580384 EC50 = 45 nM T69685 C2P4QG 44580385 EC50 = 75 nM T69685 C3UGB0 44580386 EC50 = 82 nM T69685 CE0K4J 44580471 EC50 = 46 nM T69685 CR5Y1M 44580510 EC50 > 30000 nM T69685 CBJ63S 44580511 EC50 > 30000 nM T69685 C1NME3 44580512 EC50 > 30000 nM T69685 CRCG05 44580513 EC50 > 30000 nM T69685 CMR9H1 44580514 EC50 = 52 nM T69685 CLT4V2 44580551 EC50 = 26000 nM T69685 CA92XB 44580552 EC50 = 180 nM T69685 CZK47O 44580553 EC50 = 70 nM T69685 C8YI9V 44580554 EC50 = 100 nM T69685 C54RAU 44580597 EC50 = 1600 nM T69685 CAU6P2 44580598 EC50 > 30000 nM T69685 C0PFY1 44580672 EC50 > 10000 nM T69685 C1Z8FK 44580673 EC50 = 2 nM T69685 C9KY5O 44580713 EC50 = 2 nM T69685 C52TGD 44580714 EC50 > 10000 nM T69685 CB1HZ6 44580752 EC50 = 9 nM T69685 C7L8JD 44580753 EC50 = 15 nM T69685 CB7FS6 44580754 EC50 = 69 nM T69685 C18RQM 44591636 IC50 = 5.43 nM T69685 CMTH41 44591637 IC50 = 1.74 nM T69685 C36TCP 44591639 IC50 = 124.6 nM T69685 CLO6J9 44591667 IC50 = 11.55 nM T69685 C0C1EI 44591698 IC50 = 2.95 nM T69685 CY47VM 44591699 IC50 = 3.62 nM T69685 CG3K9S 44591700 IC50 = 0.1 nM T69685 C6N7KO 44591731 IC50 = 131.7 nM T69685 CJ64OE 44591732 IC50 = 184.9 nM T69685 C0WU9E 44591733 IC50 = 870.8 nM T69685 C91NGO 44591734 IC50 = 32 nM T69685 C7B6ZT 44591763 IC50 = 0.31 nM T69685 C05LWQ 44591764 IC50 = 0.65 nM T69685 CSL6A0 44591765 IC50 = 2.58 nM T69685 CR93AQ 44591766 IC50 = 28.22 nM T69685 CFU27O 44591782 IC50 = 501.6 nM T69685 CPX59A 44591783 IC50 = 314.3 nM T69685 CQ37UV 44591785 IC50 = 123.6 nM T69685 CCA7K5 44593648 EC50 = 150 nM T69685 CZWG30 45263429 EC50 = 67 nM T69685 CT24KF 45263430 EC50 = 99 nM T69685 CSWI21 45265820 EC50 = 82 nM T69685 C14LUA 45267039 Ki = 11 nM T69685 CU0JM3 45267807 Ki = 15.2 nM T69685 CUEY48 45267808 Ki = 109 nM T69685 C18EGU 45268687 Ki = 2.32 nM T69685 CBP83E 45268691 Ki = 95.3 nM T69685 CS67XW 45270376 Ki = 3.82 nM T69685 CU4OH2 45270377 Ki = 4.58 nM T69685 CH17KU 45272913 Ki = 1.79 nM T69685 CPUR70 45272936 Ki = 2.24 nM T69685 CQ98IX 45272939 Ki = 2.32 nM T69685 C9FS6T 46213935 IC50 = 1029000 nM T69685 CL51NF 46216732 Ki = 2.5 nM T69685 CZJL95 46216733 Ki = 3.76 nM T69685 C1DO4U 46230960 Ki = 1.71 nM T69685 C59XOB 46230961 Ki = 1.98 nM T69685 C9EGU1 46230962 Ki = 2.44 nM T69685 C7G3TB 46231012 Ki = 3.96 nM T69685 C1J0WY 46231013 Ki = 5.3 nM T69685 CALC10 46231014 Ki > 641 nM T69685 C2FVA8 46231075 Ki = 2.64 nM T69685 CA3R5W 46231076 Ki = 2.9 nM T69685 CSZ2F6 46231077 Ki = 3.82 nM T69685 CVL6C0 46231146 Ki = 4.44 nM T69685 C8W4VL 46231147 Ki = 10.5 nM T69685 CRTO63 46231148 Ki = 2.79 nM T69685 CZ6C0S 46231149 Ki = 5.74 nM T69685 CTQ38S 46239398 IC50 = 25 nM T69685 C93GVI 46239399 IC50 > 10000 nM T69685 CY7S3X 46239400 IC50 = 115000 nM T69685 C4ER1X 46239401 IC50 = 112000 nM T69685 CX04CO 46239402 IC50 = 926000 nM T69685 CT14BG 46239503 IC50 = 1815000 nM T69685 CK93AJ 46239504 IC50 = 891000 nM T69685 COV4I9 46239505 IC50 = 2215000 nM T69685 CO9YC0 46239506 IC50 = 631000 nM T69685 C04GRB 46239507 IC50 = 1569000 nM T69685 C1NG0Y 46239508 IC50 = 617000 nM T69685 CC98ZF 46837246 EC50 = 80 nM T69685 C0GY1V 46837247 EC50 = 110 nM T69685 CQ41PO 46837248 EC50 = 100 nM T69685 CN1EK8 46837249 EC50 = 530 nM T69685 C5UL9K 46837250 EC50 = 900 nM T69685 CB01AC 46837364 EC50 = 80 nM T69685 C6IXU7 46837365 EC50 = 30 nM T69685 CRF5X4 46838883 EC50 > 10000 nM T69685 CVS8X0 46838884 EC50 = 9800 nM T69685 C8FZ1X 46838885 EC50 = 590 nM T69685 C6ACV2 46838886 EC50 = 34 nM T69685 CK06VF 46839028 EC50 = 18 nM T69685 C0M8AW 46839029 EC50 = 28 nM T69685 C1ZDW9 46839030 EC50 = 44 nM T69685 CZ85PM 46839031 EC50 = 390 nM T69685 C4PE5H 46839032 EC50 = 1610 nM T69685 C3L0MZ 46839160 EC50 = 500 nM T69685 C6K7FV 46839161 EC50 > 10000 nM T69685 CT51HS 46839162 EC50 = 310 nM T69685 CPI82F 46839163 EC50 = 430 nM T69685 C21ILB 46839164 EC50 = 21 nM T69685 C1OIG5 46839165 EC50 = 30 nM T69685 CB93RG 46839296 EC50 = 100 nM T69685 CS09WQ 46839297 EC50 = 91 nM T69685 C9S4IH 46839298 EC50 = 13 nM T69685 CA0MR4 46839299 EC50 = 200 nM T69685 C1EPB3 46839300 EC50 = 37 nM T69685 C57PJF 46843038 IC50 = 3 nM T69685 C0Z4TW 46848240 EC50 = 110 nM T69685 CA5KE6 46848241 EC50 = 48 nM T69685 CVU5A9 46848591 EC50 = 270 nM T69685 CJQO76 46848592 EC50 = 380 nM T69685 CNT10W 46849923 IC50 = 140 nM T69685 CH7TU9 46850094 EC50 = 24 nM T69685 CM3JH8 46850260 EC50 = 67 nM T69685 CR4OQ7 46850261 EC50 = 26 nM T69685 CWSR21 46850262 EC50 = 28 nM T69685 C28FLY 46850263 EC50 = 180 nM T69685 C2UYK7 46850264 EC50 = 10 nM T69685 CK13ZB 46850425 EC50 = 25 nM T69685 C6D9ZK 46850426 EC50 = 170 nM T69685 CFCM19 46850606 EC50 = 60 nM T69685 C48POW 46850775 EC50 = 54 nM T69685 CF8BZ4 46852151 IC50 = 1 nM T69685 CIC63B 46852155 IC50 = 78 nM T69685 CB8NF2 46852311 IC50 = 177 nM T69685 C3ZV4R 46852312 IC50 = 29 nM T69685 C9F8RE 46852316 IC50 = 211 nM T69685 CMX32J 46852462 IC50 = 18 nM T69685 CU76KJ 46852464 IC50 = 1 nM T69685 C6KZU5 46852465 IC50 = 9 nM T69685 C2Y9FU 46852773 IC50 = 3 nM T69685 C52TQR 46852924 IC50 = 340 nM T69685 CTW46S 46852926 IC50 = 946 nM T69685 CCT6Y1 46853094 IC50 = 514 nM T69685 C0U1SO 46853257 IC50 = 904 nM T69685 CAD83G 46853405 IC50 = 1703 nM T69685 CI1ES2 46853406 IC50 = 1759 nM T69685 CJ9A6U 46862338 IC50 = 58 nM T69685 CK54MW 46862340 IC50 = 2 nM T69685 CM05ZL 46862341 IC50 = 4 nM T69685 CET3L2 46862555 IC50 = 1 nM T69685 CD3I0C 46862557 IC50 = 45 nM T69685 CUL54V 46912220 IC50 = 46000 nM T69685 C40LTM 46912222 IC50 = 39000 nM T69685 C3AF9Y 46917638 IC50 > 30000 nM T69685 C2DO4V 46935693 IC50 = 627000 nM T69685 C4DJ1R 46935694 IC50 = 68000 nM T69685 CIN62E 46935749 IC50 = 40000 nM T69685 CP9JK2 46938091 IC50 = 1500000 nM T69685 C5G6IO 46938092 IC50 = 201000 nM T69685 CLC63O 46938152 IC50 = 374000 nM T69685 C5I1HQ 49798777 EC50 = 40 nM T69685 CR9N2O 52922059 IC50 > 10000 nM T69685 CF7KW0 52922061 IC50 > 10000 nM T69685 CLB47C 52922067 IC50 > 10000 nM T69685 CUY3G2 52922080 IC50 > 10000 nM T69685 CO4AW2 53317349 EC50 = 84 nM T69685 CB4J9Y 53317462 EC50 = 770 nM T69685 C2NQJ0 53318186 EC50 = 275 nM T69685 C5VTR7 53318583 EC50 = 180 nM T69685 CXY8A4 53319905 EC50 = 135 nM T69685 C65DNJ 53319906 EC50 = 805 nM T69685 C7PL6F 53319952 EC50 = 132 nM T69685 C0W2AF 53321255 EC50 = 1940 nM T69685 CO6N5I 53321256 EC50 = 250 nM T69685 C6HIS7 53322576 EC50 = 205 nM T69685 CA24UX 53323869 EC50 = 180 nM T69685 CDU0B3 53323870 EC50 = 111 nM T69685 CAM5B9 53323918 EC50 = 70 nM T69685 C89NPM 53325153 EC50 = 2080 nM T69685 CI3GU2 53325154 EC50 = 137 nM T69685 C6Y4PN 53325155 EC50 = 3000 nM T69685 C40KDP 53326450 EC50 = 2540 nM T69685 C0GT4H 53326451 EC50 = 3360 nM T69685 CQH6K5 54752777 IC50 = 79.43 nM T69685 C89ZWP 54764172 IC50 = 23.2 nM T69685 CDJ48K 54764173 IC50 = 28.1 nM T69685 CB19QJ 54764429 IC50 = 6.3 nM T69685 CNC14G 54764522 IC50 = 48.5 nM T69685 CT0F1R 54764696 IC50 = 183 nM T69685 CF0NC5 54764945 IC50 = 15.1 nM T69685 CN62OP 54764946 IC50 = 22.7 nM T69685 CH57OM 54765031 IC50 = 22 nM T69685 CE53SA 56597628 IC50 = 2.35 nM T69685 C9J7AT 56658396 IC50 = 630.96 nM T69685 CIW3R2 56658557 IC50 > 25118.86 nM T69685 CZU30J 56658558 IC50 = 2511.89 nM T69685 C2XRE3 56658559 IC50 = 501.19 nM T69685 CNY8K3 56658560 IC50 = 19952.62 nM T69685 CH73OR 56658561 IC50 = 15848.93 nM T69685 CTKI43 56658562 IC50 = 1584.89 nM T69685 CO8K7X 56659291 IC50 = 398.11 nM T69685 CXH0V2 56661885 IC50 = 3981.07 nM T69685 C1ZNL5 56662010 IC50 = 19952.62 nM T69685 C6OHX7 56662011 IC50 = 630.96 nM T69685 C89FMR 56662012 IC50 = 158.49 nM T69685 CYJ23N 56662013 IC50 = 63.1 nM T69685 C15LNY 56662014 IC50 > 25118.86 nM T69685 CHY97Q 56662751 IC50 = 1258.93 nM T69685 C9QE1S 56665356 IC50 = 10000 nM T69685 C08ALR 56665500 IC50 = 5011.87 nM T69685 CD7PK4 56665501 IC50 > 25118.86 nM T69685 CT5I3H 56665502 IC50 = 1584.89 nM T69685 C07VIA 56665503 IC50 = 19952.62 nM T69685 CG4E0X 56666222 IC50 = 63.1 nM T69685 C8HI2Y 56666223 IC50 = 1258.93 nM T69685 COR3T2 56668927 IC50 > 25118.86 nM T69685 CDM63Q 56668928 IC50 = 7943.28 nM T69685 C6QRE1 56668929 IC50 = 2511.89 nM T69685 C9HKG3 56668930 IC50 = 100 nM T69685 CA5UB3 56672410 IC50 = 15848.93 nM T69685 C6W2PY 56672411 IC50 > 25118.86 nM T69685 CU49AH 56672412 IC50 = 79.43 nM T69685 CRG5A3 56673142 IC50 = 1258.93 nM T69685 CV6FC0 56675655 IC50 = 3162.28 nM T69685 CVRC92 56676467 IC50 = 199.53 nM T69685 C9XJT7 56676468 IC50 = 1258.93 nM T69685 C1GFE0 56679109 IC50 = 6309.57 nM T69685 CGD58R 56679110 IC50 = 398.11 nM T69685 CQAZ72 56679784 IC50 = 1000 nM T69685 CAM3X5 56683113 IC50 = 1000 nM T69685 CS6GC4 56683114 IC50 = 125.89 nM T69685 C7K1FZ 57390178 IC50 = 43 nM T69685 C0XS3Y 57557326 IC50 = 39 nM T69685 CQXO18 57557335 IC50 = 1 nM T69685 C9R8MZ 57557339 IC50 = 23 nM T69685 C3UCN2 57557353 IC50 = 1 nM T69685 CIGZ78 57557375 IC50 = 16 nM T69685 C2WI3M 57557392 IC50 = 8 nM T69685 CUO9V2 58561955 IC50 = 661 nM T69685 C4D0WQ 59438392 EC50 = 660 nM T69685 CB78FY 59438397 EC50 = 180 nM T69685 C2FWT9 59438429 EC50 = 230 nM T69685 CNEJ64 59438436 EC50 = 320 nM T69685 CJ18UL 59438454 EC50 = 230 nM T69685 CGP32B 59438481 EC50 = 230 nM T69685 CO59EK 59438509 EC50 = 540 nM T69685 C3VEC7 59438510 EC50 = 670 nM T69685 C5YG1A 59438518 EC50 = 300 nM T69685 CCDQ67 66799648 IC50 = 168 nM T69685 C92QUP 66799677 IC50 = 3 nM T69685 C3H7AJ 68513937 Ki = 0.8 nM T69685 CC24FR 68943934 IC50 = 3 nM T69685 CG1O0R 70222430 IC50 = 75 nM T69685 C92VRA 70222610 IC50 = 494 nM T69685 CG1MS3 70685518 EC50 = 57 nM T69685 CY6E2Q 70691339 EC50 = 61 nM T69685 C9X7AJ 71245486 Ki = 239 nM T69685 CY7LP3 71449238 IC50 = 29 nM T69685 CZ7GW9 71452855 IC50 = 3000 nM T69685 CQ0SC1 71454631 IC50 = 7.3 nM T69685 CZ0M2C 71458193 IC50 = 3333 nM T69685 CZD12W 71458194 IC50 = 629 nM T69685 CUJT21 71582799 IC50 = 67.5 nM T69685 CVQZ85 71716253 IC50 = 782 nM T69685 CUP19I 71716254 IC50 = 175 nM T69685 C7HLS0 71716861 IC50 = 621 nM T69685 CLC3B7 71716862 IC50 = 238 nM T69685 CZHI20 71718079 IC50 = 118 nM T69685 CBL78I 71718094 IC50 = 162 nM T69685 CV2Z7K 71718685 IC50 = 523 nM T69685 C97SYX 71718694 IC50 = 4.4 nM T69685 CH5CV3 71718695 IC50 = 6400000 nM T69685 CKC70J 71719305 IC50 = 77.9 nM T69685 C72ADI 71719306 IC50 = 17.1 nM T69685 CV68AD 71719905 IC50 = 6.1 nM T69685 CA4JW0 71719906 IC50 = 2445 nM T69685 C0AIX9 71719907 IC50 = 78.4 nM T69685 CZX86Q 71719908 IC50 = 500 nM T69685 C3JAD2 71720525 IC50 = 245 nM T69685 COVM31 71720526 IC50 = 12.8 nM T69685 CJNG28 76310571 IC50 = 32 nM T69685 CND02X 76310572 IC50 = 3400 nM T69685 CD20WP 76310588 IC50 > 10000 nM T69685 CA70YQ 76310589 IC50 = 5.1 nM T69685 C2Q9WN 76310605 IC50 = 900 nM T69685 C6NST3 76314240 IC50 > 10000 nM T69685 C5YML9 76314241 IC50 > 10000000 nM T69685 C6KU8P 76317794 IC50 = 1000 nM T69685 CBR8T3 76317795 IC50 = 4 nM T69685 CG8H0J 76317812 IC50 > 10000 nM T69685 C1WVP5 76317813 IC50 = 433 nM T69685 CIO7F4 76321506 IC50 = 890 nM T69685 CJTX79 76321522 IC50 > 10000 nM T69685 CN1E8K 76321523 IC50 > 10000 nM T69685 CD2YQ8 76321524 IC50 > 10000 nM T69685 CDG09R 76325094 IC50 = 19 nM T69685 C2SM8Y 76325108 IC50 = 185000 nM T69685 C07UNT 76325109 IC50 = 64 nM T69685 C7R2YC 76325123 IC50 > 10000 nM T69685 CNIT93 76325124 IC50 = 15 nM T69685 C8YDJ5 76328661 IC50 = 82 nM T69685 CV18IA 76328662 IC50 = 1300 nM T69685 C36ULS 76328663 IC50 = 230 nM T69685 C1WEM6 76328673 IC50 = 5500 nM T69685 CZ5I8G 76328674 IC50 = 2900 nM T69685 CJ9N0S 76328675 IC50 = 247000 nM T69685 CL7J6U 76328689 IC50 = 39 nM T69685 CM23TB 76332339 IC50 = 360 nM T69685 C1S6LR 76332349 IC50 = 28 nM T69685 CV4S2L 76335970 IC50 = 100 nM T69685 C6U2PQ 76335977 IC50 > 10000 nM T69685 CN65IM 86296289 Ki = 0.002 nM T69685 CL5DH9 86296293 Ki = 0.004 nM T69685 CO02CV 86296489 Ki = 49 nM T69685 CJ57DZ 86745788 IC50 > 3000 nM T69685 CZK18W 88463909 IC50 > 10000 nM T69685 C2T4XJ 88494111 IC50 > 30000 nM T69685 CQNZ41 89621173 EC50 > 10000 nM T69685 C03GOQ 90403997 Ki = 0.029 nM T69685 CKRG60 90404317 Ki = 0.003 nM T69685 C9WC7O 90404564 Ki = 17 nM T69685 CE21TR 90404585 Ki = 0.003 nM T69685 C2DW4O 90404732 Ki = 0.118 nM T69685 C8P1SE 90404846 Ki = 0.008 nM T69685 C3DJF9 90404972 Ki = 0.199 nM T69685 CM59UR 90405129 Ki = 0.003 nM T69685 CLU6T3 90405229 Ki = 0.021 nM T69685 CXUC57 90405330 Ki = 0.093 nM T69685 CE64XQ 90405380 Ki = 198 nM T69685 CXJC03 90405436 Ki = 0.002 nM T69685 CYC82X 90405488 Ki = 0.002 nM T69685 C2JIY7 90405495 Ki = 1.25 nM T69685 CTK3H2 90405529 Ki = 0.003 nM T69685 CJHE40 90405719 Ki = 0.042 nM T69685 CF7PJ2 90405893 Ki = 1.51 nM T69685 CL1M6B 90405929 Ki = 0.06 nM T69685 CV3EU7 90406103 Ki = 0.36 nM T69685 CBY79J 90406230 Ki = 0.008 nM T69685 CHS7I5 90406432 Ki = 0.005 nM T69685 CMSC21 90406566 Ki = 0.002 nM T69685 CLY2R3 90406660 Ki = 0.007 nM T69685 C58PJY 90406771 Ki = 0.766 nM T69685 CR63IY 90406984 Ki = 1.16 nM T69685 CUN7C6 90407388 Ki = 0.005 nM T69685 C3INE9 90655881 EC50 = 1500 nM T69685 CZS60R 90655882 EC50 = 1670 nM T69685 C1OD9Y 90655883 EC50 = 1700 nM T69685 CB1RI7 90655884 EC50 = 4800 nM T69685 CLD6Z7 90655885 EC50 = 6700 nM T69685 CHZM89 90655886 EC50 = 9900 nM T69685 CKUP34 90655887 EC50 > 10000 nM T69685 CJ6N5P 90655888 EC50 > 10000 nM T69685 C8FKW1 90655889 EC50 > 10000 nM T69685 CABP58 90655890 EC50 > 10000 nM T69685 CZ76RW 90655891 EC50 > 10000 nM T69685 C01UNB 90665166 Ki = 1.79 nM T69685 C5FTW2 99116834 IC50 > 3000 nM T69685 C9ME7U 117897388 IC50 = 2.35 nM T69685 C38JEB 117897542 IC50 = 73.8 nM T69685 C3PUR8 117897549 IC50 = 2.14 nM T69685 C89EQN 117897570 IC50 = 1.03 nM T69685 CSXH08 117897680 IC50 = 1.14 nM T69685 C2ED0W 117897772 IC50 = 952 nM T69685 C5N2SK 117897780 IC50 = 56.6 nM T69685 C4A6JK 117897787 IC50 = 1.49 nM T69685 CVK03J 117897796 IC50 = 5.09 nM T69685 C30EKF 117897864 IC50 = 12.6 nM T69685 CIT13E 117897929 IC50 = 1.24 nM T69685 CU2V9L 117897938 IC50 = 8.4 nM T69685 C4CH1E 117897955 IC50 = 2294 nM T69685 CA1Z6P 117897961 IC50 = 22.7 nM T69685 CJ42DF 117897992 IC50 = 339 nM T69685 CMI40T 117898061 IC50 = 319 nM T69685 CV47YD 117898069 IC50 = 0.726 nM T69685 CGY40U 117898099 IC50 = 5.56 nM T69685 CA2L7N 117898102 IC50 = 0.671 nM T69685 CL3PM6 117898113 IC50 = 18.3 nM T69685 C7DLZ6 117898161 IC50 = 5.29 nM T69685 CO0K9G 117898177 IC50 = 0.733 nM T69685 C2U0FV 117898180 IC50 = 15.1 nM T69685 CAEK03 117898196 IC50 = 1.27 nM T69685 C2T9EV 117898210 IC50 = 5.1 nM T69685 CJB86R 117935576 IC50 > 20000 nM T69685 CS16CJ 118022791 Ki = 18 nM T69685 C89WQL 118023142 Ki = 2.6 nM T69685 CH9R8P 118023824 Ki = 44 nM T69685 CRV8S3 118478927 IC50 = 29 nM T69685 CL32JE 118478933 IC50 = 7 nM T69685 C5S1HZ 118478972 IC50 = 8 nM T69685 C8G9HP 118478986 IC50 = 113 nM T69685 CBV89G 118478994 IC50 = 23 nM T69685 CK0ER5 118478999 IC50 = 15 nM T69685 CU25KC 118479000 IC50 = 23 nM T69685 CW07IS 118479006 IC50 = 10 nM T69685 C3ZAV0 118479034 IC50 = 6 nM T69685 C4W6ZS 118479038 IC50 = 23 nM T69685 CRG24C 118479053 IC50 = 406 nM T69685 CD4ME1 118479123 IC50 = 12 nM T69685 CB0XM2 118479161 IC50 = 105 nM T69685 C18NTQ 118479199 IC50 = 55 nM T69685 CJ0Z1Y 118479222 IC50 = 441 nM T69685 CP0U6Y 118479229 IC50 = 4 nM T69685 C3A6HD 118479231 IC50 = 27 nM T69685 CJ14CR 118479241 IC50 = 38 nM T69685 C1FO3N 118479293 IC50 = 16 nM T69685 CF02TZ 118479295 IC50 = 21 nM T69685 C90TED 118479305 IC50 = 18 nM T69685 C7I9RC 118479316 IC50 = 69 nM T69685 CRC4F6 118479354 IC50 = 78 nM T69685 CRCV51 118479359 IC50 = 17 nM T69685 CJL5W0 118479428 IC50 = 12 nM T69685 CS2VA7 118479440 IC50 = 210 nM T69685 CJ9P0M 118479445 IC50 = 20 nM T69685 C3U1RB 118479452 IC50 = 10 nM T69685 CS3V4M 118937481 Ki <= 10000000 nM T69685 CXQ25D 118937486 Ki <= 100000 nM T69685 CX41RG 118937487 Ki <= 100000 nM T69685 C3S4CN 118937498 Ki <= 10000 nM T69685 CJZ94H 118937499 Ki <= 1000000 nM T69685 CF4T0E 118937507 Ki >= 10000000 nM T69685 CT9K0V 124000588 IC50 = 383 nM T69685 CTJO69 124005730 Ki = 3.3 nM T69685 COA0U2 135239967 IC50 > 30000 nM T69685 CE10YC 135239972 IC50 > 10000 nM T69685 CGEV09 135239984 IC50 > 10000 nM T69685 CY14GZ 135239991 IC50 > 10000 nM T69685 C91VJQ 135239995 IC50 > 10000 nM T69685 CL0S6Q 135240007 IC50 > 10000 nM T69685 C4E7OH 135240008 IC50 > 10000 nM T69685 C13CQX 135240011 IC50 > 30000 nM T69685 C0Q1SB 144032828 IC50 = 474 nM T69685 CC80XD 144032837 IC50 = 6 nM T69685 CN0RD7 145949219 Ki = 660 nM T69685 C18RLB 145949530 Ki = 0.097 nM T69685 CC78GK 145949682 Ki = 9.5 nM T69685 C3ASH6 145950133 Ki = 2.6 nM T69685 CXKB09 145950494 Ki = 0.9 nM T69685 CDCZ45 145950693 Ki = 0.024 nM T69685 C94NCA 145951413 Ki = 136 nM T69685 C72MQX 145952513 Ki = 1.1 nM T69685 C8M7XK 145952974 Ki = 3 nM T69685 CQG2Y3 145953118 Ki = 1.2 nM T69685 CJZ9E3 145953294 Ki = 0.001 nM T69685 C0UXK7 145953888 Ki = 141 nM T69685 C8M5HB 145956143 Ki = 2.6 nM T69685 C8RYI4 145956153 Ki = 124 nM T69685 CZVU89 145956254 Ki = 32 nM T69685 CJ8NV7 145956447 Ki = 71 nM T69685 C9C5HA 145956985 Ki = 0.8 nM T69685 CC25ZG 145957869 Ki = 1.2 nM T69685 CA1R8Y 145958038 Ki = 1.5 nM T69685 CHV19G 145959448 Ki = 1.2 nM T69685 C5ZOQ0 145959736 Ki = 3.6 nM T69685 C74NZQ 145960566 Ki = 1.2 nM T69685 C8RB9O 145962483 Ki = 5.7 nM T69685 C21LTM 145963134 Ki = 28 nM T69685 COKY15 145967585 IC50 = 7 nM T69685 CDH7S0 145968030 IC50 = 809 nM T69685 CCS80A 145968818 IC50 = 92 nM T69685 CGZ02W 145968878 IC50 = 6 nM T69685 CUR4O6 145969770 IC50 = 3362 nM T69685 CMXF86 145970099 IC50 = 1 nM T69685 CS3GE2 145970832 IC50 = 45 nM T69685 C63VEA 145971451 Ki = 69 nM T69685 CBVL78 145972216 Ki = 163 nM T69685 C5EN7V 145973394 Ki = 75 nM T69685 C6OI3K 145973962 IC50 = 10 nM T69685 CH5CL0 145974084 Ki = 35 nM T69685 C4FBU1 145986352 IC50 = 10 nM T69685 CBC0F5 154026493 IC50 > 10000 nM T69685 C16LXF 155521483 IC50 = 29 nM T69685 C10YRG 155524872 IC50 = 36.4 nM T69685 C4WJ0I 155525087 IC50 = 28.5 nM T69685 C93OTJ 155546926 IC50 = 38.4 nM T69685 CZT3W7 155547990 IC50 > 3000 nM T69685 C7NLE5 155549500 IC50 > 3000 nM T69685 CRNC68 155549901 IC50 > 3000 nM T69685 CY53JZ 155550276 IC50 > 3000 nM T69685 C1L2GT 155551564 IC50 > 3000 nM T69685 CM89BD 155555321 IC50 = 42.4 nM T69685 CGF0S6 155557862 IC50 > 3000 nM T69685 C17IVM 155558147 IC50 > 3000 nM T69685 CP2TA6 155558730 IC50 > 3000 nM T69685 C42VNF 155558759 IC50 > 3000 nM T69685 C6VDX2 155563302 IC50 > 3000 nM T69685 CA9P1T 155564998 IC50 = 9363 nM T69685 CIV8C4 155565435 IC50 = 1.54 nM T69685 C38PJX 155566448 IC50 > 3000 nM T69685 CB54HT 155568178 IC50 = 146 nM T69685 D00LNK 5311285 IC50 = 125.89 nM T69685 D07IYZ 45270374 Ki = 2.32 nM T69685 D0E1OC 16078939 IC50 = 4000 nM T69685 D0GI5V 11704260 IC50 = 3 nM T69685 D0R1ZD 59822766 IC50 = 10000 nM T69685 D0X3CF 442879 IC50 > 500000 nM T69685 D0YF9S 1088 IC50 = 91000 nM T69685 D0Z0KY 11855860 IC50 = 20 nM T76723 CWU8N7 67338 IC50 = 35000 nM T76723 CQ8A5W 91330 IC50 = 7100 nM T76723 CQEF34 1002773 IC50 > 100000 nM T76723 C89ATQ 2779831 IC50 = 19000 nM T76723 CNK84Q 7128991 IC50 > 1000000 nM T76723 CJ4IC6 24962989 IC50 > 25000 nM T76723 C0Y9FH 43199381 IC50 > 500000 nM T76723 C5N3LG 44251522 IC50 > 40000 nM T76723 C70VHB 53315882 IC50 > 10000 nM T76723 CYM2T4 53868701 IC50 > 22000 nM T76723 CPL71I 54596764 IC50 = 54000 nM T76723 CER5F1 67466175 IC50 > 100000 nM T76723 CAVD69 70678415 IC50 = 480 nM T76723 CAFU69 70686225 IC50 = 8300 nM T76723 C74BHZ 71583384 IC50 > 100000 nM T76723 C10KVQ 71583385 IC50 > 100000 nM T76723 CU6G7C 71583386 IC50 > 100000 nM T76723 C5E2IK 71583387 IC50 > 100000 nM T76723 CSX20J 71583500 IC50 > 100000 nM T76723 CS7LR9 71583501 IC50 > 100000 nM T76723 CZFG46 71583502 IC50 > 100000 nM T76723 CT64PK 71583503 IC50 > 100000 nM T76723 C10DTB 71583504 IC50 = 5900 nM T76723 CY8MN1 71583505 IC50 = 1900 nM T76723 CKN84X 71583506 IC50 = 5000 nM T76723 CZE5Q2 71583507 IC50 = 4400 nM T76723 CN0G7F 71583611 IC50 = 3300 nM T76723 CRQB87 71583612 IC50 = 490 nM T76723 CIT2D9 71583613 IC50 = 840 nM T76723 C5VN0G 71583614 IC50 = 360 nM T76723 CD7HI3 71583615 IC50 = 230 nM T76723 CVXU08 71583716 IC50 = 3600 nM T76723 C7M8OH 71583717 IC50 = 5200 nM T76723 CH0L6G 71583718 IC50 > 10000 nM T76723 C9PK2S 71583719 IC50 = 7200 nM T76723 CV03IN 71583720 IC50 > 10000 nM T76723 CAK9S7 71583721 IC50 > 50000 nM T76723 CX02GT 71583722 IC50 > 15000 nM T76723 CRJ45M 71583723 IC50 > 10000 nM T76723 C2ZY8W 71583724 IC50 > 15000 nM T76723 CIJ53B 71583833 IC50 > 15000 nM T76723 CCF58W 71583834 IC50 > 10000 nM T76723 C7N4UM 71583835 IC50 > 15000 nM T76723 CI4YA6 71583836 IC50 > 10000 nM T76723 C3C4TZ 71583837 IC50 = 300 nM T76723 CMH7J6 71583838 IC50 = 850 nM T76723 CT9Z7M 71583839 IC50 = 1800 nM T76723 CNQ73E 71583840 IC50 = 3100 nM T76723 CS3VD6 71583947 IC50 = 4000 nM T76723 CUC95I 71583948 IC50 > 25000 nM T76723 CJWU65 71583949 IC50 = 2200 nM T76723 CZ81WG 71583950 IC50 = 2700 nM T76723 C06YBC 71583951 IC50 = 3600 nM T76723 C4M7WE 71583952 IC50 = 5300 nM T76723 CJYN20 71584051 IC50 = 3300 nM T76723 C2CDB4 71716897 IC50 = 1000 nM T76723 CT85HR 71717510 IC50 > 25000 nM T76723 CF2M8S 71720569 IC50 > 100000 nM T76723 CN50PT 77620540 IC50 = 291 nM T76723 C4XJ5N 78357767 IC50 > 100000 nM T76723 C73LWN 92136227 IC50 = 4 nM T76723 CV0FW8 121225442 IC50 = 870 nM T76723 C6KV9H 124081151 IC50 > 100000 nM T76723 C2GC5B 134144476 IC50 > 28000 nM T76723 CMHQ35 134153978 IC50 = 1970 nM T76723 CB37ET 137632918 IC50 = 967 nM T76723 CK0O5H 137633979 IC50 = 833 nM T76723 CW0SC4 137634318 IC50 = 114 nM T76723 CA4N0O 137634402 IC50 = 292 nM T76723 C40XRQ 137634946 IC50 = 194 nM T76723 C4LK1X 137635057 IC50 > 50000 nM T76723 CQ2L6C 137635239 IC50 = 19 nM T76723 CQJE57 137635904 IC50 = 22 nM T76723 CSK20T 137636442 IC50 = 24 nM T76723 CKI7X0 137637621 IC50 > 50000 nM T76723 C7LYB4 137638165 IC50 > 1900 nM T76723 CYF9N2 137638943 IC50 = 22 nM T76723 CV0FG8 137642089 IC50 = 2594 nM T76723 CLN3Q6 137642237 IC50 = 35 nM T76723 C1LS6B 137643074 IC50 = 757 nM T76723 CBF5W9 137644102 IC50 > 5000 nM T76723 CV7F1Q 137644278 IC50 = 150 nM T76723 CRX70A 137644349 IC50 = 84 nM T76723 CF4G2Z 137645564 IC50 = 46 nM T76723 CQW2K9 137645780 IC50 = 87 nM T76723 CJW1C5 137646449 IC50 > 2000 nM T76723 C0G2JH 137646885 IC50 = 295 nM T76723 CGYX94 137647553 IC50 = 477 nM T76723 C4NZ2E 137648946 IC50 > 8000 nM T76723 C6DM5E 137649738 IC50 = 17 nM T76723 CS4AU2 137650745 EC50 = 1600 nM T76723 CTLX12 137651083 IC50 = 158 nM T76723 CN7EP0 137651766 IC50 = 10 nM T76723 CENR64 137654339 IC50 = 36 nM T76723 CRT8Q3 137655207 IC50 = 22 nM T76723 CXI7M3 137656669 IC50 = 421 nM T76723 CPEZ15 137657265 IC50 = 55 nM T76723 C7BH1Z 137658189 IC50 = 1938 nM T76723 CA53WC 137660734 IC50 = 476 nM T76723 C7DUV4 137660840 IC50 = 166 nM T76723 C7N6LE 137661325 IC50 = 61 nM T76723 CDPN65 137661881 IC50 > 50000 nM T76723 C7LI1Z 137662076 IC50 = 540 nM T76723 CR5D4S 138753329 IC50 = 3000 nM T76723 C51ILK 138753330 IC50 = 15000 nM T76723 CE58DF 153041236 IC50 > 100000 nM T76723 C7C8HI 155529624 IC50 > 10000 nM T76723 CJ8ZI6 155549992 IC50 > 200000 nM T76723 D00JWB 90642938 IC50 = 19 nM T76723 D02TVQ 71268957 IC50 = 74000 nM T76723 D09CLP 439155 IC50 = 2000 nM T76723 D0AF1J 53346504 IC50 = 1600 nM T76723 D0BU8W 44219611 IC50 > 25000 nM T76723 D0CX4W 46901937 IC50 > 40000 nM T76723 D0L0DC 53339032 Ki = 1150 nM T76723 D0Q3FY 44622850 IC50 > 25000 nM T70840 D0E6XR 3062316 IC50 = 114 nM T70840 D09XZL 56962369 IC50 = 24 nM T70840 D0E3TC 44259 IC50 = 2.44 nM T70840 D03BNU 59604787 IC50 > 10000 nM T70840 CZ0T5U 2948 IC50 = 800 nM T70840 CO1HN4 237073 IC50 > 100000 nM T70840 CFZW70 258149 IC50 = 4000 nM T70840 CW6Z3E 290232 IC50 = 4400 nM T70840 C3OH1T 318013 IC50 = 4300 nM T70840 CY9U5J 323535 IC50 > 100000 nM T70840 CU9MA5 336250 IC50 > 100000 nM T70840 C0ZKD5 337817 IC50 > 100000 nM T70840 CAS18T 359052 IC50 = 37000 nM T70840 CL1JC9 405801 IC50 = 5300 nM T70840 C5Q4VB 433561 IC50 > 100000 nM T70840 CB7RL2 600546 IC50 > 100000 nM T70840 CR98MZ 613528 IC50 = 9000 nM T70840 CL5PU0 650805 IC50 = 12700 nM T70840 CP2QJ7 660775 IC50 = 4000 nM T70840 C7PMQ2 676971 IC50 > 100000 nM T70840 C3JVL2 716205 IC50 = 3000 nM T70840 CL3B8P 723159 IC50 > 100000 nM T70840 C3SPC8 731510 IC50 > 100000 nM T70840 CW6RH8 738893 IC50 > 100000 nM T70840 C84ZOX 765847 IC50 = 56000 nM T70840 CFB5G4 766178 IC50 = 7100 nM T70840 CV9US2 789677 IC50 = 2800 nM T70840 CR0EW6 826476 IC50 > 100000 nM T70840 C4LS3M 830964 IC50 > 100000 nM T70840 CWF41G 832424 IC50 > 100000 nM T70840 C5W8XA 863538 IC50 > 100000 nM T70840 CDHN42 888669 IC50 = 11000 nM T70840 C07CXM 911790 IC50 = 1600 nM T70840 C28XAY 939263 IC50 = 41000 nM T70840 CW7H0Z 1005440 IC50 = 1300 nM T70840 CYP8Z3 1006295 IC50 = 30000 nM T70840 CR8DA2 1008507 IC50 = 44000 nM T70840 CX34GM 1391336 IC50 = 2000 nM T70840 C6ZY1V 1641261 IC50 > 100000 nM T70840 CX95WT 2270285 IC50 > 100000 nM T70840 CV29EU 2736849 IC50 > 100000 nM T70840 CQ1S0O 2740613 IC50 = 2500 nM T70840 CZQ87D 2791276 IC50 > 100000 nM T70840 C9T1RS 2881040 IC50 > 100000 nM T70840 CSD3F2 3116802 IC50 = 18000 nM T70840 C0E3QB 3161284 IC50 > 100000 nM T70840 C7HP0V 3724764 IC50 > 100000 nM T70840 C2VI5M 4112641 IC50 > 100000 nM T70840 CO3WS1 5008522 IC50 = 700 nM T70840 C8Q4WH 8027126 IC50 > 100000 nM T70840 CS19YL 10104270 IC50 = 7000 nM T70840 C8G3UE 10805474 IC50 = 37000 nM T70840 CBOP58 11293798 Ki > 10000 nM T70840 C26BZX 11362471 Ki > 10000 nM T70840 CWXB93 11397177 Ki > 10000 nM T70840 CTG83F 11539329 Ki > 9600 nM T70840 CMIL86 11590363 Ki > 9600 nM T70840 C9T6SC 11640926 Ki > 9600 nM T70840 CE1T7R 12353991 IC50 = 15000 nM T70840 C1VY5X 13793449 IC50 = 92000 nM T70840 CX7O3M 14513911 IC50 = 660 nM T70840 CFPW41 16007116 Ki > 9500 nM T70840 CA7CR3 16069860 IC50 = 2700 nM T70840 CJ9I2T 25190908 IC50 = 9000 nM T70840 CC71QJ 27666048 IC50 = 3200 nM T70840 C2QCX6 41316396 IC50 > 100000 nM T70840 CN8WB9 44189332 IC50 = 36 nM T70840 CRZ79W 44542926 IC50 = 3.7 nM T70840 CE0O4B 44543079 IC50 = 6.6 nM T70840 CQT48I 44543080 IC50 = 3.2 nM T70840 C3VRO9 44557921 IC50 > 10000 nM T70840 CM3GX4 45102613 IC50 = 18 nM T70840 C0FM5X 45381385 IC50 = 43 nM T70840 C7J0OL 45381386 IC50 = 315 nM T70840 CY3HW5 46224684 IC50 = 4700 nM T70840 CD2K4R 50908681 IC50 = 759000 nM T70840 CV0CZ5 52942728 IC50 = 252 nM T70840 CIVE91 52949671 IC50 = 4.01 nM T70840 CHK60J 54680213 IC50 > 100000 nM T70840 CL54GO 56660026 IC50 = 4000 nM T70840 CN6CP2 56660027 IC50 = 2800 nM T70840 CYX48O 56663445 IC50 = 1800 nM T70840 C7VSF1 56663493 IC50 = 3500 nM T70840 CAT1K4 56666872 IC50 = 9500 nM T70840 CI0XD1 56666922 IC50 = 300 nM T70840 C15DPN 56666923 IC50 = 2300 nM T70840 CFP8L2 56666924 IC50 > 20000 nM T70840 CC4KQ9 56670364 IC50 = 9100 nM T70840 C18TIU 56670365 IC50 > 20000 nM T70840 CX6H3R 56673818 IC50 = 2100 nM T70840 C58BWU 56673867 IC50 = 17000 nM T70840 C6WZK4 56683837 IC50 = 260 nM T70840 CHB41Q 56683838 IC50 = 3200 nM T70840 C2PO7W 56683839 IC50 = 11000 nM T70840 CS9TY6 56683840 IC50 = 8600 nM T70840 C7LAS5 56965901 IC50 = 10 nM T70840 CR2ZM0 57391854 IC50 > 10000 nM T70840 CF89DG 57398808 IC50 > 10000 nM T70840 C4DM3N 57398809 IC50 > 10000 nM T70840 CTJI57 57404047 IC50 = 201 nM T70840 CI1A8M 57404048 IC50 = 62 nM T70840 CPGR16 57404049 IC50 > 10000 nM T70840 CO7SX4 57920205 IC50 = 19 nM T70840 C3V6MX 57920210 IC50 = 134 nM T70840 CI50KU 58167984 IC50 = 18 nM T70840 C86YRV 58688296 IC50 = 227 nM T70840 C8AT5N 58688313 IC50 = 145 nM T70840 C09YWX 58688317 IC50 = 172 nM T70840 C4Q2HL 58688342 IC50 = 284 nM T70840 C0LK4S 58688380 IC50 = 32 nM T70840 CF4S6Q 58688403 IC50 > 50000 nM T70840 CNVK41 58688409 IC50 = 163 nM T70840 CJI0Q4 58688436 IC50 = 210 nM T70840 CK1AO4 58688444 IC50 = 38 nM T70840 CZ0J6F 58688467 IC50 = 1663 nM T70840 CPE98M 58688474 IC50 = 359 nM T70840 CDOK25 58688484 IC50 = 444 nM T70840 CHO5G0 58688561 IC50 = 115 nM T70840 CP2JK1 58688569 IC50 = 64 nM T70840 CIV53P 58688575 IC50 = 23 nM T70840 CVO46Z 58688633 IC50 = 368 nM T70840 C2T8UL 58688642 IC50 = 213 nM T70840 CP9N3K 62705016 IC50 = 55 nM T70840 C14CUM 65629114 IC50 > 100000 nM T70840 C3IZ0N 66548972 IC50 = 87 nM T70840 CA3Y4X 66549150 IC50 > 1000 nM T70840 CJ4SC2 66549151 IC50 = 145 nM T70840 CQWF78 66549338 IC50 = 78 nM T70840 CJWM52 66549339 IC50 = 237 nM T70840 CKW80R 66549342 IC50 = 1600 nM T70840 CENC12 66549526 IC50 = 2400 nM T70840 C13EIQ 66549529 IC50 = 120 nM T70840 C3JZN9 66549530 IC50 = 156 nM T70840 C7ECR3 66549904 IC50 = 81 nM T70840 CSJ2O4 66549905 IC50 = 228 nM T70840 CEO7I8 66550128 IC50 = 44 nM T70840 C6QE0Z 66550129 IC50 = 395 nM T70840 C4H7LO 66550130 IC50 = 181 nM T70840 C3EPF1 66550131 IC50 = 230 nM T70840 C07AMS 66550133 IC50 = 149 nM T70840 C0H9SX 66550353 IC50 = 204 nM T70840 C0YSI4 66550560 IC50 = 196 nM T70840 C0AS4Z 66550763 IC50 = 172 nM T70840 CT94GU 66550766 IC50 = 159 nM T70840 CS7N8U 66550768 IC50 = 361 nM T70840 CT48BH 66550769 IC50 = 5700 nM T70840 CG5RL3 66550770 IC50 = 5500 nM T70840 CK2L8N 66550966 IC50 = 795 nM T70840 CZ85QK 66551165 IC50 = 732 nM T70840 CT1C4Z 66551562 IC50 = 379 nM T70840 C21CHX 66551563 IC50 = 498 nM T70840 CV63UL 67240318 IC50 > 10000 nM T70840 CF9PI3 68386640 IC50 = 231 nM T70840 C5RPF7 68518614 IC50 = 80 nM T70840 C78YUA 68518851 IC50 = 35 nM T70840 C50YAE 68520214 IC50 > 10000 nM T70840 CNIM41 68520578 IC50 = 283 nM T70840 C2VOK4 68521168 IC50 = 710 nM T70840 CDM0U9 68521184 IC50 = 142 nM T70840 C3T6GU 68522253 IC50 = 1527 nM T70840 CE3A0Q 68522320 IC50 = 85 nM T70840 C8B5YJ 68522434 IC50 = 75 nM T70840 CTJ23Y 69495841 IC50 = 4000 nM T70840 CIJ5L9 70682556 IC50 = 250 nM T70840 C9IB8C 70684645 IC50 = 87 nM T70840 CH08ZN 70690951 IC50 = 1037 nM T70840 C9SU2M 70697187 IC50 = 485 nM T70840 CK0CH3 70697188 IC50 = 12500 nM T70840 C5NR6E 70812853 IC50 = 828 nM T70840 CH5QO0 70812854 IC50 = 50 nM T70840 CGS60U 70812857 IC50 = 4100 nM T70840 C91WQB 70812860 IC50 = 199 nM T70840 C2J8UX 70812861 IC50 > 1000 nM T70840 C60GRO 70812863 IC50 = 998 nM T70840 C9BT7J 70812868 IC50 = 6100 nM T70840 CA10BZ 70812876 IC50 = 129 nM T70840 C2AHO7 70812880 IC50 = 127 nM T70840 CU9L5N 70812942 IC50 = 243 nM T70840 C3J6MB 70812946 IC50 = 223 nM T70840 C3TOI5 70812989 IC50 = 294 nM T70840 CDE3C1 71038721 IC50 = 34000 nM T70840 CT92OL 71295837 IC50 = 80 nM T70840 CF87LR 71449511 IC50 = 43000 nM T70840 C8R5VS 71451313 IC50 > 100000 nM T70840 CKT60L 71455860 Ki = 194 nM T70840 CZM1K4 71765510 IC50 = 12 nM T70840 C0DL3F 72698602 IC50 = 1.74 nM T70840 CB5MP3 87482409 IC50 = 203 nM T70840 CU6P2V 88992379 IC50 = 310 nM T70840 C7UXE0 90659701 IC50 = 4 nM T70840 CXT56Y 90666099 IC50 = 43000 nM T70840 C12CTW 90666100 IC50 > 50000 nM T70840 C1E6PA 91938057 IC50 = 23 nM T70840 C9R3XZ 102532131 IC50 = 58 nM T70840 CCRI64 102532132 IC50 = 19 nM T70840 CR8J5P 116812154 IC50 = 19000 nM T70840 CBO67F 117908368 IC50 = 15 nM T70840 CE1U4R 117908383 IC50 = 270 nM T70840 CNS7E5 117908420 IC50 = 3100 nM T70840 CK2DP0 117918816 IC50 = 9200 nM T70840 C36YMI 117918825 IC50 = 20 nM T70840 C6R9IK 117918840 IC50 = 500 nM T70840 CI6CT8 117918855 IC50 = 2200 nM T70840 CO2A6W 117918867 IC50 = 5 nM T70840 CV4RL7 117918880 IC50 = 2500 nM T70840 C7S8DX 117918881 IC50 = 3 nM T70840 C62ATU 117918908 IC50 = 574 nM T70840 CO2KG8 117918912 IC50 = 82 nM T70840 CAM1V7 117918913 IC50 = 120 nM T70840 CTLS12 117918919 IC50 = 8 nM T70840 CH4GF2 117918922 IC50 = 1 nM T70840 CRDS25 117918940 IC50 = 3300 nM T70840 CJC26Z 117918945 IC50 = 850 nM T70840 C0X2OP 117918947 IC50 = 327 nM T70840 CW5Y4R 117918955 IC50 = 620 nM T70840 C06HGS 117918979 IC50 = 3 nM T70840 C1Z5CX 118718090 IC50 = 220 nM T70840 C5LXS9 118718094 IC50 = 376 nM T70840 CXWM35 118718095 IC50 = 163 nM T70840 C24BIT 118732089 IC50 = 60 nM T70840 CTJZ54 118732090 IC50 = 4507 nM T70840 CLQB81 118732091 IC50 = 368 nM T70840 CI38QT 118732092 IC50 = 132 nM T70840 C1VES6 118732093 IC50 = 101 nM T70840 CH3ZB0 118732094 IC50 = 86 nM T70840 CSYA60 118732095 IC50 = 67 nM T70840 C0K5LC 118732096 IC50 = 25 nM T70840 C8UN3S 118732097 IC50 = 350 nM T70840 CW2ZV1 118732098 IC50 = 151 nM T70840 C4HM7F 118732099 IC50 = 37 nM T70840 C5QTK1 118732100 IC50 = 913 nM T70840 C41IOQ 118732101 IC50 = 100 nM T70840 C2R9JZ 118732102 IC50 = 53 nM T70840 C8VL9G 118732103 IC50 = 27 nM T70840 CZO5W1 118732104 IC50 = 21 nM T70840 C0KG9I 118732105 IC50 = 47 nM T70840 CR1Z0O 118732106 IC50 = 20 nM T70840 C4IQ7C 118732107 IC50 = 21 nM T70840 CSLU37 118732108 IC50 = 21 nM T70840 CYRJ23 118732109 IC50 = 8 nM T70840 CL8WE1 118732110 IC50 = 1090 nM T70840 CLD74V 118732111 IC50 = 9240 nM T70840 CCA4U3 118732112 IC50 > 10000 nM T70840 C1ACJ0 122189152 IC50 = 16 nM T70840 CTOX13 122189153 IC50 = 27 nM T70840 CA0NQ6 122189154 IC50 = 18 nM T70840 CXK73S 122189155 IC50 = 37 nM T70840 CUYA85 122189156 IC50 = 38 nM T70840 CQS34F 122189157 IC50 = 57 nM T70840 CE13UV 122189158 IC50 = 41 nM T70840 C4E8IF 122189159 IC50 = 50 nM T70840 CCT83H 122189160 IC50 = 41 nM T70840 CY23RV 122189161 IC50 = 50 nM T70840 CFJR29 122189162 IC50 = 7.6 nM T70840 CEX47Y 122189163 IC50 = 23 nM T70840 CUB9Q5 122189164 IC50 = 282 nM T70840 C63OQZ 122189165 IC50 = 65 nM T70840 CG51VB 122189166 IC50 = 1000 nM T70840 CH74JB 122189167 IC50 = 31 nM T70840 C0SO5F 122189168 IC50 > 1000 nM T70840 CUML53 122189169 IC50 = 945 nM T70840 C23PWJ 122189170 IC50 > 1000 nM T70840 C4M6BZ 122189171 IC50 = 239 nM T70840 C5ZO6J 122189172 IC50 > 10000 nM T70840 C36LON 122189173 IC50 = 25 nM T70840 C5IDL1 122189174 IC50 = 20 nM T70840 CTQ9U7 122189175 IC50 = 23 nM T70840 C31YGS 122189176 IC50 = 26 nM T70840 CC48FJ 122189177 IC50 = 22 nM T70840 CV2U0H 122192497 IC50 = 6600 nM T70840 CDN7R2 122192498 IC50 >= 30000 nM T70840 C9Y0PI 122194166 IC50 = 10 nM T70840 C0C4EH 122194167 IC50 = 11 nM T70840 C03GHF 122194168 IC50 = 19 nM T70840 CT56LG 122194169 IC50 = 55 nM T70840 CZ7CJ6 127047267 IC50 = 18 nM T70840 CAW6X5 127047919 IC50 = 22 nM T70840 C3YE1D 127048049 IC50 = 22 nM T70840 C2QP4D 127048050 IC50 = 20 nM T70840 C3B4HT 136003186 IC50 = 7732 nM T70840 CZ1U5T 136265485 IC50 = 267 nM T70840 CE9CU2 136265599 IC50 = 571 nM T70840 C6XIE9 136624922 IC50 = 260 nM T70840 C6L3HN 137634634 IC50 = 44 nM T70840 C2MD1Q 155513187 IC50 > 10000 nM T70840 D00ERW 44444843 Ki > 9546 nM T70840 D00HVA 11624601 Ki > 9600 nM T70840 D03PVS 821974 IC50 = 33000 nM T70840 D07XWC 44477445 IC50 = 0.5 nM T70840 D0F6NZ 58688690 IC50 = 66 nM T70840 D0FC4Y 46192505 IC50 = 1 nM T70840 D0Q3NG 11715520 Ki > 9600 nM T70840 D0S0XD 58688563 IC50 = 30 nM T70840 D0S7IE 11658882 Ki > 9600 nM T70840 D0US9O 45275255 IC50 = 63 nM T45674 D01ZSO 4235 Ki > 200 nM T45674 D0D1AL 3559 Ki = 16 nM T45674 D0H2SE 118607347 Ki = 48 nM T45674 D0W3TS 41306362 Ki = 190 nM T45674 D0XK2K 9829526 Ki = 0.12 nM T45674 C7B8VJ 44405080 Ki = 1550 nM T45674 CLY10I 65659 Ki > 200 nM T45674 CI8KD2 97627 Ki = 796 nM T45674 CS4XQ9 1081502 Ki > 200 nM T45674 C6Z4QI 3050372 Ki = 25.1 nM T45674 C5NA6S 3069135 Ki = 5.12 nM T45674 C6AX8Y 3126148 Ki > 200 nM T45674 C4Z0DT 9049339 Ki = 160 nM T45674 CTAC24 9885114 Ki = 231 nM T45674 CZ9MG4 10356384 Ki > 200 nM T45674 C5F4WP 10403711 Ki = 4350 nM T45674 CC1AT3 11165837 Ki = 10.33 nM T45674 CBFZ60 11531451 Ki = 113 nM T45674 C1HDM5 11653679 Ki = 5.129 nM T45674 CCG14E 13091356 Ki = 18 nM T45674 CYN95Z 13091359 Ki = 29 nM T45674 C65SCN 15599151 Ki = 432 nM T45674 CTME96 16202156 Ki = 0.26 nM T45674 C45JHX 17644936 Ki > 200 nM T45674 C7MST8 17758676 Ki = 12.6 nM T45674 CCM1L3 18118650 Ki = 340 nM T45674 CZ31UL 18118651 Ki > 1200 nM T45674 C9UE6C 18118654 Ki > 1200 nM T45674 CWQ5S7 27148262 Ki = 360 nM T45674 C4MRQ0 27842480 Ki = 2750 nM T45674 CUVS17 29048070 Ki = 95 nM T45674 C7EJK2 31588412 Ki = 321 nM T45674 CO9HV7 40624141 Ki > 1200 nM T45674 CRJ5E1 41306333 Ki > 1200 nM T45674 CCF93H 41306385 Ki = 350 nM T45674 CQSO71 41306434 Ki > 1200 nM T45674 CGO25K 41306445 Ki = 310 nM T45674 C83TBP 41307231 Ki = 200 nM T45674 CK5Z6Q 45160790 Ki = 1995.26 nM T45674 C3A9OY 51111240 Ki = 470 nM T45674 CPJZ31 52149645 Ki = 200 nM T45674 C82HKM 52750322 Ki = 160 nM T45674 CIW0F6 54582640 Ki = 227 nM T45674 CZU6L2 57345618 Ki = 5.888 nM T45674 CK9G8H 57345619 Ki = 8.5 nM T45674 C4EXS6 57396571 Ki = 33 nM T45674 CYN38R 57401819 Ki = 51.5 nM T45674 C3TNQ5 60346448 Ki = 850 nM T45674 C7JG9R 60701380 Ki > 400 nM T45674 C7FMA4 70676458 Ki = 2010 nM T45674 C28RIZ 76518514 Ki = 25.12 nM T45674 CLM0J5 90644067 Ki = 600 nM T45674 CH5R8Q 98049507 Ki = 32 nM T45674 CO6Z7J 110440208 Ki = 200 nM T45674 CBW0U9 110445832 Ki = 98 nM T45674 CHU07G 118607283 Ki = 170 nM T45674 CX2QI6 118607309 Ki = 1400 nM T45674 CIW02L 118607351 Ki = 200 nM T45674 C84QJX 118607364 Ki = 59 nM T45674 CX5B2A 118607439 Ki = 170 nM T45674 CXOT38 118607453 Ki = 49 nM T45674 C4U2GB 118607455 Ki = 20 nM T45674 CSB25E 118709750 Ki = 8.1 nM T45674 CD4S9R 118709751 Ki = 2.138 nM T45674 CM57GR 126720252 Ki = 1200 nM T45674 CN91JP 137632351 Ki = 8.4 nM T45674 CUV20T 137636134 Ki = 76.1 nM T45674 C4PAF3 137642542 Ki = 22.3 nM T45674 C5NL4A 137645149 Ki = 23 nM T45674 C92HOT 137650821 Ki = 23.8 nM T45674 C6GZR2 137653169 Ki = 24 nM T45674 CM7IN4 137657904 Ki = 16.2 nM T45674 CZG4P7 137662176 Ki = 25.5 nM T45674 C1TQ2A 145953153 Ki = 110 nM T45674 CXEV63 145954849 Ki = 5.19 nM T45674 CDGA65 145956728 Ki = 350 nM T45674 CJA9T4 146597626 Ki > 10000 nM T45674 C3D4UM 146597628 Ki > 10000 nM T45674 C7UHR0 146597630 Ki = 251.19 nM T45674 CCRS21 146597638 Ki > 10000 nM T45674 CM18OU 146597639 Ki = 630.96 nM T45674 C42TIZ 146597651 Ki = 398.11 nM T45674 CL5PG8 146597666 Ki > 10000 nM T45674 C89YUC 146597677 Ki > 10000 nM T45674 CU9G0O 146597678 Ki > 10000 nM T45674 C6TRC9 146641556 Ki > 10000 nM T45674 C8I3YJ 146641558 Ki = 100 nM T45674 C3LBA0 146641564 Ki > 10000 nM T45674 CFD4N9 146641568 Ki = 501.19 nM T45674 CP70WA 146641787 Ki > 10000 nM T45674 C0WU5Y 146641788 Ki > 10000 nM T45674 C10LOP 146641795 Ki = 251.19 nM T45674 CG97ER 146709966 Ki = 316.23 nM T45674 C6FX4M 147636204 Ki = 1000 nM T45674 CW4S2X 147652368 Ki > 10000 nM T45674 CF5B2L 147653864 Ki = 630.96 nM T45674 C5PNX8 148302367 Ki = 316.23 nM T45674 C2E5HK 149396365 Ki = 100 nM T45674 C9T0PS 153061504 Ki = 1995.26 nM T45674 CF7J3M 153287535 Ki = 3981.07 nM T45674 C72MVW 153287537 Ki = 1258.93 nM T45674 CAF36V 153287539 Ki = 79.43 nM T45674 C1FA0K 153287541 Ki = 316.23 nM T45674 CEQ69Z 153287542 Ki = 125.89 nM T45674 C9A7SV 153287550 Ki > 10000 nM T45674 C91KST 153287551 Ki = 1258.93 nM T45674 C6P3SR 153287553 Ki = 1000 nM T45674 C3G5CJ 153287557 Ki = 79.43 nM T45674 CW31CT 153287566 Ki = 158.49 nM T45674 CYP86E 153287567 Ki = 316.23 nM T45674 CS73ZC 153287568 Ki = 316.23 nM T45674 CV9G7Z 153287572 Ki > 10000 nM T45674 CO85KL 153287574 Ki = 630.96 nM T45674 CCD9N1 155512086 Ki = 753 nM T45674 CTV8R1 155512151 Ki = 642 nM T45674 CV35ZN 155513505 Ki = 662 nM T45674 C2D8ZF 155515129 Ki = 7.61 nM T45674 C58EAT 155515524 Ki = 11 nM T45674 C5K2GQ 155516317 Ki = 14 nM T45674 C4KWA1 155518665 Ki = 2.512 nM T45674 CUSA24 155519891 Ki > 10000 nM T45674 CU8D3T 155519913 Ki = 16 nM T45674 CIP3X7 155523942 Ki = 21.8 nM T45674 CY17EB 155524132 Ki = 4.6 nM T45674 CY5Q0J 155524744 Ki = 11 nM T45674 C9W2NV 155525645 Ki = 158.49 nM T45674 CP76JX 155526977 Ki > 10000 nM T45674 CW6CX1 155528147 Ki = 1673 nM T45674 CPA51T 155528865 Ki = 42.66 nM T45674 C3Z5XG 155529711 Ki = 7.6 nM T45674 C8RGT9 155532745 Ki = 5.5 nM T45674 CV83SG 155534733 Ki = 1720 nM T45674 C7PO3B 155535411 Ki = 64.1 nM T45674 C7PW0N 155535978 Ki = 8 nM T45674 CB79ZW 155536080 Ki > 10000 nM T45674 CIUS98 155536619 Ki = 2090 nM T45674 CR16NT 155540848 Ki = 39.81 nM T45674 CW76ES 155542765 Ki = 87 nM T45674 CMT60C 155543832 Ki = 349 nM T45674 CIA1C9 155547197 Ki = 32 nM T45674 CJ1U4N 155547337 Ki = 16 nM T45674 CF7MQ8 155550094 Ki > 10000 nM T45674 CI41QF 155552117 Ki = 2550 nM T45674 CJ92EA 155552895 Ki = 316.23 nM T45674 CKSZ39 155553997 Ki = 13 nM T45674 C04OFL 155554079 Ki = 2.2 nM T45674 CRU26E 155554287 Ki = 125.89 nM T45674 CZ9U5N 155554849 Ki = 251.19 nM T45674 C5EVM7 155555743 Ki = 651.6 nM T45674 CC48RQ 155556295 Ki = 25.12 nM T45674 CBS89O 155556618 Ki = 1170 nM T45674 CJBX01 155557042 Ki = 3162.28 nM T45674 C8TO2W 155558029 Ki = 1300 nM T45674 C4QID8 155558857 Ki = 6.7 nM T45674 CK4Z6D 155559218 Ki = 7.9 nM T45674 C4J0ZI 155559223 Ki > 10000 nM T45674 C13RCK 155561279 Ki = 13.1 nM T45674 CXYQ73 155561471 Ki = 31.62 nM T45674 CCOD50 155562467 Ki = 1980 nM T45674 C4N9GU 155563428 Ki = 2020 nM T45674 CK9RN6 155563452 Ki = 8.4 nM T45674 CSM7V1 155564110 Ki = 7.943 nM T45674 CR0F6E 155565622 Ki = 68.8 nM T45674 CBI7N3 155566272 Ki = 583 nM T45674 CNCT72 155568142 Ki = 3.8 nM T45674 C5N2EK 155568367 Ki > 1000 nM T45674 D02WJT 7333 Ki = 20 nM T45674 D0F0IA 11301655 Ki > 2000 nM T45674 D0KL1P 10474335 Ki = 0.34 nM T45674 D0P0XA 197060 Ki = 90.4 nM T45674 D0Q7FM 15443 Ki = 50.12 nM T88304 D09FAZ 9444 IC50 = 300 nM T88304 D0U5SI 4913 IC50 > 500000 nM T88304 D0X5XU 451668 IC50 = 30 nM T88304 D0L4FS 5280961 IC50 = 30000 nM T88304 D0U2BH 65064 IC50 = 500 nM T88304 D02VTV 117968550 EC50 = 100000 nM T88304 D03LZO 117967861 EC50 = 46000 nM T88304 C5IO2D 171251 IC50 > 45000 nM T88304 CKS4U8 188380 IC50 = 302000 nM T88304 CJH6D9 327606 IC50 = 100000 nM T88304 CA6J0D 445762 IC50 = 18000 nM T88304 C3KVN2 702558 IC50 = 390000 nM T88304 CQEF34 1002773 IC50 > 100000 nM T88304 CJ4ID2 3718032 IC50 = 12000 nM T88304 CG0D6N 10451940 IC50 > 100000 nM T88304 CZC4W3 11576752 IC50 = 27000 nM T88304 CIC81U 21120307 IC50 = 45000 nM T88304 CDMU19 24828467 IC50 = 150000 nM T88304 C85NAQ 24858111 IC50 = 850 nM T88304 C2ENB5 24947577 IC50 = 18000 nM T88304 C6D0LY 30118838 IC50 = 20000 nM T88304 CW7Z9B 45267108 IC50 = 6000 nM T88304 CBYR03 45267109 IC50 = 31000 nM T88304 C4YJQ9 45267958 IC50 > 10000 nM T88304 CYBW25 45267964 IC50 = 216000 nM T88304 CR4BF6 45267973 IC50 = 7400 nM T88304 CL0JD3 45267974 IC50 = 820 nM T88304 C70YFN 45267975 IC50 = 36000 nM T88304 CGYV47 45267981 IC50 = 22000 nM T88304 CP1OF8 45268848 IC50 = 75000 nM T88304 C7T2ZU 45268859 IC50 = 5000 nM T88304 CT84RL 45269774 IC50 > 100000 nM T88304 CX6H5T 45270517 IC50 = 8000 nM T88304 CE7K6J 45270523 IC50 = 154000 nM T88304 CR5B0C 45270527 IC50 = 5400 nM T88304 C54CSO 45270528 IC50 = 3700 nM T88304 C90XJH 45270533 IC50 = 6700 nM T88304 C6YIP2 45270600 IC50 = 8000 nM T88304 CK8BR2 45271342 IC50 = 44000 nM T88304 CCV8K1 45271353 IC50 = 44000 nM T88304 CHE5I6 45271416 IC50 > 100000 nM T88304 CQP6C4 45271423 IC50 = 300000 nM T88304 C87VSU 45272236 IC50 = 2500 nM T88304 CWD34S 45272237 IC50 = 4500 nM T88304 C2PUO3 45272238 IC50 = 4800 nM T88304 CL19VE 45272250 IC50 = 15000 nM T88304 CZJ86D 45272318 IC50 > 100000 nM T88304 CD47UG 45272319 IC50 = 4000 nM T88304 C83FZD 45273085 IC50 = 45000 nM T88304 C2YXN3 45273086 IC50 = 2900 nM T88304 C5MO1Y 45273087 IC50 = 21000 nM T88304 CDJE90 45273088 IC50 > 100000 nM T88304 CRE09G 45273096 IC50 = 19000 nM T88304 CWO9X2 45273097 IC50 = 94000 nM T88304 CIX92D 45273102 IC50 = 61000 nM T88304 C7E9SW 45273103 IC50 = 2500 nM T88304 CN96GS 45273186 IC50 = 1100 nM T88304 C03YWX 49786972 Ki > 50000 nM T88304 CPL71I 54596764 IC50 = 121000 nM T88304 CFY18X 56643471 IC50 = 150000 nM T88304 C32POU 56648592 IC50 = 270000 nM T88304 C0IPV6 56648595 IC50 = 1600000 nM T88304 C2AP8B 56648690 IC50 = 570000 nM T88304 CXBY54 56648693 IC50 = 310000 nM T88304 CQ34RM 56648770 IC50 = 1130000 nM T88304 C0XFZ5 56935564 IC50 = 4000 nM T88304 CJBY70 56951879 IC50 = 2.9 nM T88304 CB49HN 59457966 IC50 = 173000 nM T88304 C7M0FJ 59457983 IC50 = 370 nM T88304 CER5F1 67466175 IC50 > 100000 nM T88304 CO3F1Q 70686507 IC50 = 22000 nM T88304 C62WVR 70695988 IC50 = 132000 nM T88304 C9NV1Z 76310239 IC50 = 98000 nM T88304 CJ8H5F 76310241 IC50 = 40000 nM T88304 C52YJT 76310995 IC50 = 4110 nM T88304 CD1M0Q 76313934 IC50 = 20000 nM T88304 CNQ86R 76314627 IC50 = 174000 nM T88304 CAKL96 76314628 IC50 = 68000 nM T88304 CYB1U4 76318201 IC50 = 9000 nM T88304 C18MDV 76321200 IC50 = 80000 nM T88304 CZ09ML 76321898 IC50 = 35000 nM T88304 CF3KG5 76325534 IC50 = 38600 nM T88304 C4OYL7 76325535 IC50 = 27900 nM T88304 C08QPM 76328372 IC50 = 73000 nM T88304 CFX2B7 76328373 IC50 = 230000 nM T88304 CA54DX 76332046 IC50 = 128000 nM T88304 C84NAS 76332047 IC50 = 50000 nM T88304 CY05NB 76332742 IC50 = 12300 nM T88304 CDL08Z 76336365 IC50 = 650 nM T88304 C4XJ5N 78357767 IC50 > 100000 nM T88304 C01DAP 86288828 IC50 = 179000 nM T88304 CVM64R 117967504 EC50 = 30000 nM T88304 CJY5W0 117967660 EC50 = 73000 nM T88304 CM5N2A 117967691 EC50 = 27000 nM T88304 C2G4ND 117967705 EC50 = 26000 nM T88304 CY1V9T 117976066 EC50 = 32000 nM T88304 CY2R4J 117976176 EC50 = 20000 nM T88304 CSTY10 118607373 IC50 = 73 nM T88304 C9BI8F 118607414 IC50 = 619 nM T88304 CSW92P 118607432 IC50 = 382 nM T88304 CO1D7I 118607435 IC50 = 4420 nM T88304 C6PZ1X 118607459 IC50 = 750 nM T88304 CBA79J 118607465 IC50 = 645 nM T88304 CLS25W 118607471 IC50 = 494 nM T88304 C1K0VJ 118607474 IC50 = 1370 nM T88304 C8XMV5 118607488 IC50 = 497 nM T88304 CY1X2K 118613614 IC50 = 950 nM T88304 CT6OD8 118613615 IC50 = 1070 nM T88304 COPW27 118613616 IC50 > 10000 nM T88304 CJW05H 118613617 IC50 = 978 nM T88304 C7X2AQ 118613624 IC50 = 413 nM T88304 CE69HN 118613626 IC50 = 297 nM T88304 CDK3F2 118613628 IC50 = 1080 nM T88304 C5AF9V 118613631 IC50 = 1050 nM T88304 CG39ZR 118613632 IC50 = 582 nM T88304 CUDE80 118613633 IC50 = 969 nM T88304 CLIZ07 118613634 IC50 = 230 nM T88304 CG6E0J 118613636 IC50 = 1050 nM T88304 C07LSQ 118613637 IC50 = 1410 nM T88304 CB0K3S 118613639 IC50 = 232 nM T88304 C7SIL0 118613641 IC50 = 1250 nM T88304 CQD69N 118613646 IC50 = 234 nM T88304 CQNA84 118613647 IC50 = 201 nM T88304 CBC0Q9 118613651 IC50 = 290 nM T88304 C2EQ9X 118613653 IC50 = 140 nM T88304 C1X8GW 118613658 IC50 = 123 nM T88304 C0JVC9 118613660 IC50 = 957 nM T88304 CI70WP 118613691 IC50 = 316.23 nM T88304 CQ5T3E 118613693 IC50 > 10000 nM T88304 CFGK68 118613694 IC50 = 618 nM T88304 C1LOF4 118613696 IC50 = 759 nM T88304 CAY5Q6 118613697 IC50 = 1600 nM T88304 CG7D9I 118613701 IC50 = 945 nM T88304 C3ZJO5 118613702 IC50 = 2290 nM T88304 COJB60 118613705 IC50 = 929 nM T88304 CX8J7D 118613718 IC50 = 1270 nM T88304 CKI70Y 118613722 IC50 = 624 nM T88304 CJY8E1 118613723 IC50 = 781 nM T88304 CPW12K 118613724 IC50 = 1030 nM T88304 C3QX6D 118613726 IC50 = 137 nM T88304 CKO15P 118613728 IC50 = 1790 nM T88304 CW1D6K 118613729 IC50 = 32 nM T88304 CGQ82T 118732749 IC50 = 19000 nM T88304 CV0FW8 121225442 IC50 = 150 nM T88304 C6G0CZ 122580323 EC50 > 100000 nM T88304 CJI14M 129072680 IC50 = 21 nM T88304 CU3FP1 129072681 IC50 = 83 nM T88304 C0ES4L 129072695 IC50 = 588 nM T88304 COL81P 129085358 IC50 = 40 nM T88304 CUZ6K0 129085359 IC50 = 2080 nM T88304 CI1H4A 129085361 IC50 = 298 nM T88304 C2B5VP 129085364 IC50 = 274 nM T88304 CJ18GA 129085365 IC50 = 247 nM T88304 CUO5E6 129085366 IC50 = 425 nM T88304 CVPH43 129085367 IC50 = 212 nM T88304 CKS08I 129085368 IC50 = 446 nM T88304 CNO1K2 129085369 IC50 = 414 nM T88304 CIST32 129085377 IC50 = 200 nM T88304 CL9KB8 129246684 IC50 = 1870 nM T88304 C6ZYB8 129270457 IC50 = 1320 nM T88304 CL0WR7 134386479 EC50 > 100000 nM T88304 C5H9YP 135398693 IC50 > 1000000 nM T88304 C6GC0O 137028680 EC50 > 100000 nM T88304 C4S1ZI 137333995 IC50 = 3100 nM T88304 CWMH49 137638632 EC50 = 16000 nM T88304 C05DFP 137653852 EC50 = 24000 nM T88304 C95RGF 145950703 IC50 = 231 nM T88304 C0XBU5 145951018 IC50 = 284 nM T88304 CIKY95 145954902 IC50 = 2250 nM T88304 C5NS1C 145963999 IC50 = 475 nM T88304 CMX3R9 145964677 IC50 = 722 nM T88304 C7XF6P 145965645 IC50 = 501 nM T88304 CW2ZV7 145967174 IC50 = 80 nM T88304 C39OCT 145967367 IC50 = 494 nM T88304 C3JO8Q 145971403 IC50 = 187 nM T88304 COJG25 145974212 IC50 = 261 nM T88304 CKVI47 145974419 IC50 = 83 nM T88304 CW1LX9 145975217 IC50 = 235 nM T88304 CIP42V 145976082 IC50 = 211 nM T88304 C8MFK6 145977537 IC50 = 205 nM T88304 C5I0ZL 145977690 IC50 = 833 nM T88304 CU2A1M 145978072 IC50 = 234 nM T88304 C3MF6X 145978745 IC50 = 250 nM T88304 CUVO30 155515610 EC50 > 100000 nM T88304 CX5G9E 155528619 EC50 > 100000 nM T88304 CS3PF1 155533577 EC50 > 100000 nM T88304 CRH9J5 155534178 EC50 > 100000 nM T88304 CAE51Q 155534378 EC50 > 100000 nM T88304 C29RHJ 155544579 EC50 > 100000 nM T88304 CIN57Q 155556138 IC50 = 14000 nM T88304 CB8SD4 155557649 EC50 > 100000 nM T88304 C0BU1J 155560963 EC50 > 100000 nM T88304 D02TVQ 71268957 IC50 > 100000 nM T88304 D06PPL 25150857 IC50 > 10000 nM T88304 D07VWC 344265 IC50 = 50000 nM T88304 D08TGQ 124349 IC50 = 1500 nM T88304 D09CLP 439155 IC50 = 4000 nM T88304 D0A2ZH 266989 IC50 = 212000 nM T88304 D0BI4T 53315878 IC50 > 50000 nM T88304 D0GK7A 46224516 IC50 = 1287 nM T88304 D0I2RW 8342 IC50 = 1600 nM T88304 D0J5VK 67145 IC50 = 47000 nM T88304 D0L0DC 53339032 Ki = 950 nM T88304 D0S9SJ 56962337 IC50 = 0.3 nM T89917 D04AIT 5280445 IC50 = 20000 nM T89917 D07EXH 359 IC50 > 200000 nM T89917 D07MGA 72281 IC50 = 8300 nM T89917 D0J9ZR 4477 IC50 = 40000 nM T89917 D0K8KX 5280343 IC50 = 8100 nM T89917 C5H9TY 14697 IC50 = 207000 nM T89917 C3I7VB 102678 IC50 = 24500 nM T89917 CL5Y4J 159516 Ki = 3100 nM T89917 CV0B7W 442027 IC50 = 49600 nM T89917 C1E2FR 442048 IC50 = 283500 nM T89917 CZ3MD8 647122 IC50 = 16100 nM T89917 C2C8QU 948801 Ki = 27500 nM T89917 CXA4P6 1265413 IC50 = 90720 nM T89917 CUD4A1 1328543 IC50 = 58350 nM T89917 C3ZP4U 2131972 Ki = 9110 nM T89917 CA1N3H 2131982 Ki = 9930 nM T89917 CKL8B2 2219105 IC50 = 29900 nM T89917 CN43XQ 2806068 IC50 = 160 nM T89917 C5J6MO 2849659 IC50 = 28800 nM T89917 CN3P7A 2911959 IC50 = 74500 nM T89917 CZDG23 2947583 IC50 = 186000 nM T89917 CBIP72 2986413 IC50 = 76700 nM T89917 CCU3P7 3635406 IC50 = 2200 nM T89917 CZF0R5 4004950 IC50 = 500 nM T89917 C3AN7C 4117477 IC50 = 1180 nM T89917 CS2WB7 4236803 IC50 = 29800 nM T89917 C0AW3N 4378077 IC50 = 13860 nM T89917 CO3Y0T 4614896 IC50 = 9910 nM T89917 CY68ZT 4788586 IC50 = 940 nM T89917 CTR4Q1 5320532 IC50 = 13300 nM T89917 CVG47I 5958938 IC50 = 10500 nM T89917 CD8ZT2 6026688 IC50 > 50000 nM T89917 C3LZX9 8027611 IC50 = 12660 nM T89917 CJ4C5K 9180583 IC50 = 10800 nM T89917 CYQ8Z4 9882716 IC50 > 50000 nM T89917 C8K2NO 10062715 IC50 = 800000 nM T89917 C49CMU 10411574 IC50 = 21700 nM T89917 C6GN2F 11642725 IC50 = 870000 nM T89917 CHYP53 12310492 IC50 = 233400 nM T89917 C65EOH 15949840 IC50 = 7500 nM T89917 C9V8EM 15956553 IC50 = 300000 nM T89917 C3WYR4 16061499 IC50 = 2000 nM T89917 CTO43V 16085283 Ki = 116000 nM T89917 CU35DQ 21582568 IC50 = 220800 nM T89917 CN45FL 23427055 IC50 = 164700 nM T89917 CK3AF8 25256829 IC50 = 5400 nM T89917 C2SZ7L 42624533 IC50 = 14000 nM T89917 CYP8V1 44404067 IC50 > 50000 nM T89917 CD20PF 44433696 IC50 = 80000 nM T89917 CI4P2V 44433697 IC50 = 10000 nM T89917 CW7B0J 44433698 IC50 = 15000 nM T89917 C8DWL3 44433699 IC50 = 200000 nM T89917 C0ZPE2 44517748 IC50 = 2700 nM T89917 C0OH2T 44584893 IC50 = 5400 nM T89917 C0NZ5E 44584944 IC50 = 7300 nM T89917 CT70DZ 44590821 IC50 = 22500 nM T89917 C0SW2K 45266425 IC50 = 2500 nM T89917 C5WBP2 45266482 IC50 = 3800 nM T89917 CA4K8F 45266488 IC50 = 6600 nM T89917 C3BHZ4 45268445 IC50 > 50000 nM T89917 CC05NI 45268452 IC50 = 15400 nM T89917 C6QD9E 45269292 IC50 > 50000 nM T89917 CY7RV4 45269761 Ki = 21000 nM T89917 CO80TH 45269762 Ki = 297000 nM T89917 CU34ZK 45269763 Ki = 584000 nM T89917 C9P3LZ 45269764 Ki = 478000 nM T89917 CXS19V 45269765 Ki = 45200 nM T89917 C3DY4T 45270971 IC50 > 50000 nM T89917 CR4WA8 45270979 IC50 = 20900 nM T89917 CM78GO 45271412 Ki = 462000 nM T89917 CC90BU 45271826 IC50 = 5200 nM T89917 C0B6KX 45271831 IC50 = 9300 nM T89917 CN85IQ 45271832 IC50 = 8100 nM T89917 C7IF2O 45272299 Ki = 363000 nM T89917 CZRV73 45272304 Ki = 34100 nM T89917 CGV14L 45272305 Ki = 112000 nM T89917 CVTL97 45272306 Ki = 2200 nM T89917 CAM89I 45273174 Ki = 135000 nM T89917 CZT67B 45273179 Ki = 614000 nM T89917 CHF4M5 45273180 Ki = 49300 nM T89917 CND1R3 45273184 Ki = 159000 nM T89917 C0V5WT 45273625 IC50 > 50000 nM T89917 C6OE7V 46784066 IC50 = 28300 nM T89917 C6LH5I 46881919 Ki = 800 nM T89917 CI2FO1 49870840 IC50 = 5500 nM T89917 CF2D0I 49870841 IC50 = 8400 nM T89917 CM52SZ 49870842 IC50 = 6800 nM T89917 C8Q2CZ 50885062 IC50 > 50000 nM T89917 CJ6KV7 52941131 IC50 = 13900 nM T89917 C8M2QD 52943127 IC50 = 24300 nM T89917 CQ84MD 52945913 IC50 = 12000 nM T89917 CJ1LG2 52945915 IC50 = 42000 nM T89917 CZ35DX 52945977 IC50 = 128900 nM T89917 CAB1Y3 52946772 IC50 = 163200 nM T89917 CO4R1B 52947200 IC50 = 18000 nM T89917 CC4X1O 52948928 IC50 = 137700 nM T89917 CMG4U7 52949213 IC50 = 10800 nM T89917 C0X5BL 58589722 IC50 = 76740 nM T89917 CY3CL6 71544384 IC50 = 610 nM T89917 CV3P2U 71544385 IC50 = 230 nM T89917 CJS60O 71571220 IC50 = 49000 nM T89917 C1AY0M 71571221 IC50 = 49000 nM T89917 CY21XB 71571222 IC50 = 4600 nM T89917 C1DX9H 71571223 IC50 = 39000 nM T89917 CKE2C3 73056463 IC50 > 100000 nM T89917 C9S8ZH 73056464 IC50 > 100000 nM T89917 CK9OI0 73056465 IC50 = 31710 nM T89917 C4D8LK 73056466 IC50 = 32080 nM T89917 CRY86G 73056467 IC50 = 34910 nM T89917 C3VS4F 73056760 IC50 = 10070 nM T89917 CYH1F4 73056761 IC50 = 51330 nM T89917 C2CRZ8 73056762 IC50 = 2250 nM T89917 CD4YR3 73056763 IC50 = 11830 nM T89917 C3P2OZ 73056764 IC50 = 67200 nM T89917 C1H8PX 73056765 IC50 = 82910 nM T89917 C8JO7B 73056766 IC50 = 13860 nM T89917 CCYE63 73057087 IC50 = 5520 nM T89917 C54JWM 73057088 IC50 = 39870 nM T89917 C8RBU6 73057089 IC50 = 1040 nM T89917 CEBH65 73057090 IC50 = 1690 nM T89917 C8M2DX 73057091 IC50 = 17820 nM T89917 CQ42AZ 73057092 IC50 = 2820 nM T89917 CPLJ64 73057388 IC50 = 4700 nM T89917 CIN5V0 76320984 IC50 = 4300 nM T89917 C05AYV 102341658 IC50 = 16400 nM T89917 C8S3CR 102341659 IC50 = 37500 nM T89917 C2G9CP 127043455 IC50 = 20200 nM T89917 CVZ4I3 127043641 IC50 = 6000 nM T89917 C7BST4 127043642 IC50 = 5800 nM T89917 CGO01F 127043643 IC50 > 50000 nM T89917 C2TU5A 127043644 IC50 = 6400 nM T89917 C0Y9IT 127043645 IC50 = 41200 nM T89917 CF3B1Z 127045220 IC50 = 11700 nM T89917 CIXJ94 127045221 IC50 = 8600 nM T89917 CQ1CT5 127045222 IC50 = 18700 nM T89917 CKRX04 127045227 IC50 = 30700 nM T89917 CDZ2E1 127045228 IC50 > 50000 nM T89917 CG3E9B 127045229 IC50 = 6700 nM T89917 CG6VR3 127045386 IC50 = 15700 nM T89917 CK9JE3 127045387 IC50 > 50000 nM T89917 CY1E4Z 127045392 IC50 > 50000 nM T89917 CK5PA4 127045393 IC50 = 44700 nM T89917 C34TWD 127045394 IC50 > 50000 nM T89917 C97MQC 127048409 IC50 = 20000 nM T89917 C41VRM 127048410 IC50 = 7500 nM T89917 CZ0B1R 127052510 IC50 = 10000 nM T89917 CRW05E 127052511 IC50 > 50000 nM T89917 CC3TX0 127052512 Ki = 72000 nM T89917 CIQ1U9 127052513 Ki = 41000 nM T89917 CI13JZ 135452883 IC50 = 10000 nM T89917 CG1KW5 135470831 IC50 = 77090 nM T89917 CH4Q6A 145964401 IC50 = 5500 nM T89917 CHU61S 145964420 IC50 = 42100 nM T89917 C6YCA8 145964710 IC50 = 28800 nM T89917 CV6F7L 145966788 IC50 = 2100 nM T89917 CBWX17 145967285 IC50 = 4300 nM T89917 COR9X3 145972736 IC50 = 3900 nM T89917 CQ0M2X 145972809 IC50 = 4100 nM T89917 CF95RZ 145972878 IC50 = 3200 nM T89917 CXI0D1 145975081 IC50 = 6300 nM T89917 CG84ZR 145975487 IC50 = 5100 nM T89917 C91FOT 145976006 IC50 = 5200 nM T89917 C3F4UH 145978039 IC50 = 8800 nM T89917 CL7FB0 2919450 IC50 = 62790 nM T89917 D00RIX 5280443 IC50 = 280800 nM T89917 D01XMM 4117383 IC50 = 4450 nM T89917 D08MZY 145937 Ki = 8200 nM T89917 D08UYP 3008868 Ki = 2400 nM T89917 D09BUG 10207 IC50 = 132000 nM T89917 D0L7AT 10480940 Ki = 19300 nM T89917 D0S0BN 130976 Ki = 10600 nM T89917 D0SY2M 5281708 IC50 = 105000 nM T89917 D0UQ6U 10569 IC50 = 189100 nM T89917 D0WA9S 10429214 IC50 = 146500 nM T65501 C5IO2D 171251 IC50 = 17000 nM T65501 CF8YA5 442757 IC50 = 500 nM T65501 CA6J0D 445762 IC50 = 41000 nM T65501 CZC4W3 11576752 IC50 = 2000 nM T65501 CBX8T9 16451230 IC50 > 200000 nM T65501 CIC81U 21120307 IC50 = 6800 nM T65501 C85NAQ 24858111 IC50 = 7500 nM T65501 C2ENB5 24947577 IC50 = 900 nM T65501 CW7Z9B 45267108 IC50 = 1000 nM T65501 CBYR03 45267109 IC50 = 21000 nM T65501 CYBW25 45267964 IC50 = 500000 nM T65501 CR4BF6 45267973 IC50 = 600 nM T65501 CL0JD3 45267974 IC50 = 1900 nM T65501 C70YFN 45267975 IC50 > 45000 nM T65501 CGYV47 45267981 IC50 = 3600 nM T65501 C7T2ZU 45268859 IC50 = 27000 nM T65501 CT84RL 45269774 IC50 = 39000 nM T65501 CX6H5T 45270517 IC50 = 3000 nM T65501 CE7K6J 45270523 IC50 = 2000 nM T65501 CR5B0C 45270527 IC50 = 600 nM T65501 C54CSO 45270528 IC50 = 260 nM T65501 C90XJH 45270533 IC50 = 29000 nM T65501 C6YIP2 45270600 IC50 = 1500 nM T65501 CK8BR2 45271342 IC50 = 26000 nM T65501 CCV8K1 45271353 IC50 > 100000 nM T65501 CHE5I6 45271416 IC50 = 54000 nM T65501 CQP6C4 45271423 IC50 = 28000 nM T65501 C87VSU 45272236 IC50 = 6800 nM T65501 C2PUO3 45272238 IC50 = 12000 nM T65501 CL19VE 45272250 IC50 = 33000 nM T65501 CZJ86D 45272318 IC50 > 100000 nM T65501 C83FZD 45273085 IC50 = 45000 nM T65501 C2YXN3 45273086 IC50 = 57200 nM T65501 C5MO1Y 45273087 IC50 = 256000 nM T65501 CDJE90 45273088 IC50 = 11000 nM T65501 CRE09G 45273096 IC50 = 100000 nM T65501 CWO9X2 45273097 IC50 = 66000 nM T65501 CIX92D 45273102 IC50 = 1000 nM T65501 C7E9SW 45273103 IC50 = 920 nM T65501 CN96GS 45273186 IC50 = 300 nM T65501 CIZF42 122178085 IC50 > 50000 nM T65501 C5H9YP 135398693 IC50 > 1000000 nM T65501 D08TGQ 124349 IC50 = 300 nM T65501 D09CLP 439155 IC50 = 200 nM T65501 D0J5VK 67145 IC50 = 17000 nM T40097 D0EG1I 9926791 IC50 > 10000 nM T40097 D0J9ZR 4477 IC50 > 100000 nM T40097 D02UFQ 11620908 IC50 > 10000 nM T40097 D05ADP 160355 IC50 = 170000 nM T40097 D0E3TC 44259 IC50 = 361 nM T40097 D0HY9S 73386890 IC50 = 92 nM T40097 D0O6ZO 9952773 IC50 > 10000 nM T40097 D0Q7RE 16007391 Ki > 10000 nM T40097 D0S6TK 11213558 EC50 = 10 nM T40097 D0X4MN 11597537 Ki = 44 nM T40097 D03BNU 59604787 IC50 > 10000 nM T40097 D05SJB 10040667 IC50 = 101 nM T40097 D08DNZ 45102739 IC50 = 14 nM T40097 D08JIS 46926788 IC50 = 1300 nM T40097 D09QKG 25104303 EC50 = 10100 nM T40097 D0ID4H 2190145 IC50 = 26000 nM T40097 D0PG5N 25123232 IC50 = 7780 nM T40097 D0UY9Y 46869000 IC50 = 220 nM T40097 D0W7MG 11647397 IC50 = 1100 nM T40097 D0W8BL 46868926 IC50 = 2 nM T40097 D0X7OF 46926710 IC50 = 2700 nM T40097 D0ZU8L 57340689 IC50 = 1.3 nM T40097 D04WCI 16220188 IC50 = 5420 nM T40097 D0A9KI 9863367 IC50 > 50 nM T40097 D0H4GI 10275001 IC50 = 448 nM T40097 D0T3ME 156422 IC50 > 10000 nM T40097 CJ17AM 4877 IC50 = 270 nM T40097 COYW98 9222 IC50 > 667000 nM T40097 CW3VJ0 55970 IC50 = 48 nM T40097 C9W4UM 290221 IC50 > 10000 nM T40097 C3V0TX 447873 IC50 = 2 nM T40097 C9VW8M 449054 IC50 > 16000 nM T40097 CKG76T 579429 IC50 > 10000 nM T40097 CQ9PB5 684674 IC50 > 10000 nM T40097 CK89TF 766948 IC50 > 10000 nM T40097 CHRN50 854156 Ki = 2060 nM T40097 CKS84B 897877 IC50 = 800 nM T40097 CIHE37 905354 IC50 > 100000 nM T40097 C3PBJ1 942437 IC50 > 50000 nM T40097 CO0S8U 971337 IC50 = 3162.28 nM T40097 C6K8WV 979869 IC50 = 360 nM T40097 C4XP1N 1100747 IC50 > 10000 nM T40097 CRGB47 1228713 IC50 > 100000 nM T40097 C67OWG 1228882 IC50 > 100000 nM T40097 C78JFC 1246652 IC50 = 1400 nM T40097 C7ALK5 1246796 IC50 = 2900 nM T40097 C0SLP9 1489193 IC50 > 10000 nM T40097 C6F7JZ 2090652 IC50 = 11900 nM T40097 CPM53W 2091135 IC50 > 25000 nM T40097 C1DSP5 2114077 IC50 = 18700 nM T40097 CL32PJ 2126205 IC50 = 9400 nM T40097 CCG85A 2128371 IC50 > 50000 nM T40097 CNB6D2 2137680 IC50 > 100000 nM T40097 C5VE3K 2231029 IC50 = 2100 nM T40097 C2S4ZO 2311248 IC50 = 15400 nM T40097 CSD8C9 2377140 IC50 = 5700 nM T40097 C72CNT 2747117 IC50 = 280 nM T40097 CZHL80 2808202 IC50 = 1600 nM T40097 C65FZH 2970548 IC50 > 100000 nM T40097 CNG1X0 2971028 IC50 = 5900 nM T40097 C9WJE0 3656000 IC50 = 6700 nM T40097 C8WSF5 3659633 IC50 = 12500 nM T40097 C0D3PQ 4018929 IC50 > 25000 nM T40097 CR0DJ8 4078145 IC50 > 100000 nM T40097 C69GSP 4079571 IC50 = 700 nM T40097 C2GS6L 4146014 IC50 = 8400 nM T40097 CE2M9B 5066795 IC50 = 1600 nM T40097 C4BC3G 6104220 IC50 > 100000 nM T40097 CA32PV 6540289 IC50 = 1220 nM T40097 C38UZJ 6852206 IC50 = 77 nM T40097 COY61K 7164065 IC50 > 100000 nM T40097 C3O0NW 7164103 IC50 = 5400 nM T40097 C5X4ES 7167021 IC50 = 3600 nM T40097 C4EJ6T 7597300 IC50 = 5100 nM T40097 CMK84C 8719932 IC50 = 1900 nM T40097 C5H4VR 8867965 IC50 = 2800 nM T40097 CX5FW7 8903993 IC50 > 50000 nM T40097 C3JEN8 9543521 IC50 = 230 nM T40097 CSFQ07 9549178 IC50 = 101 nM T40097 C4Z2GW 9819930 IC50 > 10000 nM T40097 C1E2DV 9826083 IC50 = 1500 nM T40097 CRC65X 9863786 IC50 > 10000 nM T40097 CJ4QV2 9885993 IC50 = 16000 nM T40097 CHF7G5 9890746 IC50 > 30000 nM T40097 CS5P9X 9890933 IC50 = 34 nM T40097 C3EUB4 9911005 IC50 > 30000 nM T40097 CX5G3A 9928616 IC50 = 5350 nM T40097 C0V7UW 9958506 IC50 = 30 nM T40097 CQP98N 10002079 IC50 = 850 nM T40097 C26QHZ 10005638 IC50 > 10000 nM T40097 C93OCY 10021870 IC50 = 780 nM T40097 C7YD1X 10048045 IC50 > 25000 nM T40097 C4PRY1 10066845 IC50 = 42 nM T40097 CF1D6Y 10075240 IC50 > 10000 nM T40097 CLA50K 10091293 IC50 = 261 nM T40097 CPN3T4 10092520 IC50 = 106 nM T40097 C9NO1X 10149689 IC50 = 1600 nM T40097 CYE4T2 10151272 IC50 = 698 nM T40097 CN0QK4 10152189 IC50 = 228 nM T40097 C76HSI 10153026 IC50 = 9.2 nM T40097 C69DHW 10158652 IC50 < 16000 nM T40097 CR47IV 10172440 IC50 = 246 nM T40097 CT4X3K 10195059 IC50 = 9.6 nM T40097 C7QHS0 10215642 IC50 = 61 nM T40097 C1I0SL 10247954 IC50 = 384 nM T40097 C9JB7R 10289046 IC50 = 20 nM T40097 C7SFI1 10296883 IC50 > 10000 nM T40097 CB59MP 10310219 IC50 = 45 nM T40097 CFL5O8 10364826 IC50 = 88 nM T40097 CA8B5T 10390073 IC50 = 1900 nM T40097 C95LYF 10457505 IC50 > 30000 nM T40097 CB0E2X 10472936 IC50 = 451 nM T40097 CJ4P5T 10905857 IC50 > 30000 nM T40097 CT7N3S 11213972 IC50 = 6.4 nM T40097 CA36OM 11236353 IC50 = 398.11 nM T40097 C2AG5I 11257276 IC50 = 794.33 nM T40097 CWY63O 11269297 IC50 = 501.19 nM T40097 CBOP58 11293798 Ki > 10000 nM T40097 C26BZX 11362471 Ki > 10000 nM T40097 C1G4UY 11372308 IC50 = 15.85 nM T40097 CK26AG 11374509 IC50 = 794.33 nM T40097 CWXB93 11397177 Ki > 10000 nM T40097 C0APW4 11422034 IC50 = 150 nM T40097 CI5XE7 11463002 IC50 = 125.89 nM T40097 C9TKF0 11476467 IC50 = 794.33 nM T40097 C1W7UV 11486202 IC50 = 199.53 nM T40097 C7UVM8 11492814 IC50 > 10000 nM T40097 CH6XL5 11493316 IC50 = 400 nM T40097 CRS89T 11499625 IC50 = 310 nM T40097 CCV71Z 11500561 IC50 = 420 nM T40097 CXBU49 11502255 IC50 = 385000 nM T40097 CU0QR2 11509379 IC50 = 1700 nM T40097 CY20KH 11514465 IC50 = 1400 nM T40097 CLC92Y 11514477 IC50 > 10000 nM T40097 C7H6PZ 11516913 IC50 = 69 nM T40097 CJ9OH7 11538129 IC50 = 320 nM T40097 CTG83F 11539329 Ki = 3 nM T40097 C4U3YQ 11543503 IC50 = 4800 nM T40097 CJ97XP 11544489 IC50 = 580 nM T40097 CF7JG0 11551231 IC50 = 510 nM T40097 CM57ZU 11553156 IC50 = 69 nM T40097 C7DX5S 11558435 IC50 = 260 nM T40097 C5VML9 11558444 IC50 > 10000 nM T40097 C4I0YH 11558900 IC50 = 210 nM T40097 C3KT8X 11559766 IC50 = 74 nM T40097 CVS32L 11560956 IC50 = 28 nM T40097 C70ROB 11564900 IC50 = 910 nM T40097 C78ZTX 11565848 IC50 = 2600 nM T40097 CK9D6M 11579435 IC50 > 10000 nM T40097 C9XBP4 11580158 IC50 = 2700 nM T40097 CYK05Q 11586583 IC50 = 2400 nM T40097 C6O0HX 11587896 IC50 = 120 nM T40097 C24JGU 11589125 IC50 = 110 nM T40097 CQ82SM 11589163 IC50 = 87 nM T40097 CMIL86 11590363 Ki = 3 nM T40097 C4S3JZ 11600899 IC50 = 2200 nM T40097 CB59ND 11601122 IC50 > 10000 nM T40097 CZ70BL 11601246 IC50 = 4000 nM T40097 CVH94J 11601374 IC50 = 8900 nM T40097 CUK87R 11602023 IC50 = 190 nM T40097 CQ29WV 11602291 IC50 = 180 nM T40097 C7TXB8 11609198 IC50 = 270 nM T40097 C1A4SV 11615890 IC50 = 350 nM T40097 C73PTY 11616278 IC50 = 6300 nM T40097 C5B3XJ 11620410 IC50 > 40000 nM T40097 COT15X 11622644 IC50 > 10000 nM T40097 CFD43W 11624410 IC50 = 3500 nM T40097 CSM62L 11626920 IC50 > 30000 nM T40097 C9NP0W 11638309 IC50 = 290 nM T40097 CSNY14 11638719 IC50 > 10000 nM T40097 C9T6SC 11640926 Ki = 1 nM T40097 C6NO5B 11647280 IC50 = 35 nM T40097 C5ENI8 11651832 IC50 = 890 nM T40097 C9VP4Y 11655237 IC50 = 37 nM T40097 CX1T5L 11666890 IC50 = 300 nM T40097 CKDU79 11666971 IC50 = 4400 nM T40097 C4CF9O 11667089 IC50 = 300 nM T40097 CV6Y3Z 11673227 IC50 > 10000 nM T40097 C9GN5Y 11674342 IC50 = 1100 nM T40097 CR1WD2 11678117 IC50 = 8.2 nM T40097 CY5TR4 11680140 IC50 > 10000 nM T40097 CJ9KN7 11683817 IC50 > 10000 nM T40097 CU0E8O 11690457 Ki > 2000 nM T40097 C2CPZ3 11695458 IC50 = 160 nM T40097 C9I7QG 11697773 IC50 = 400 nM T40097 CM1KG9 11705144 IC50 = 3000 nM T40097 CB0AP2 11705863 Ki > 10000 nM T40097 C9P0VD 11729539 IC50 > 30000 nM T40097 CD7IZ6 11785059 IC50 = 158.49 nM T40097 CBC08P 11846124 IC50 = 4.7 nM T40097 CD60CH 11846125 IC50 = 12 nM T40097 C5LIW2 11846126 IC50 = 26 nM T40097 CNJB87 11846287 IC50 = 4 nM T40097 CEMS06 11846288 IC50 = 6400 nM T40097 C7DI3U 11846294 IC50 = 390 nM T40097 CVS03I 11846457 IC50 > 10000 nM T40097 CX8B0G 11846458 Ki = 400 nM T40097 CIJ93W 11846459 IC50 = 71 nM T40097 C5KC7Q 11846461 IC50 = 270 nM T40097 CAZS08 11848309 IC50 > 10000 nM T40097 C43IVN 11848567 IC50 > 10000 nM T40097 C9LAY8 11848825 IC50 > 10000 nM T40097 CC09DE 11955790 IC50 = 10500 nM T40097 CEX45S 12723726 IC50 = 2800 nM T40097 C09ERV 14555267 IC50 = 3162.28 nM T40097 CGFP41 14617322 IC50 = 6800 nM T40097 CYFH12 15658026 IC50 = 7700 nM T40097 CBF4X2 15991561 IC50 > 10000 nM T40097 CFPW41 16007116 Ki = 3.8 nM T40097 C9TU1O 16046126 IC50 > 1000 nM T40097 C3V6EX 16049812 IC50 = 15 nM T40097 CZHJ34 16058637 IC50 = 9 nM T40097 CKR57M 16086104 IC50 > 10000 nM T40097 C16NRY 16086114 IC50 = 389 nM T40097 C5VPH9 16129448 IC50 = 82 nM T40097 C0C5AZ 16129582 IC50 = 13 nM T40097 C6L9VD 16216351 IC50 = 23 nM T40097 CR7J3V 16230198 IC50 = 65300 nM T40097 CM6IG4 16231644 IC50 = 75100 nM T40097 C3EUA0 16362025 IC50 = 6200 nM T40097 CU56EW 16664858 IC50 > 10000 nM T40097 CAG75U 16849419 IC50 > 25000 nM T40097 C7MLQ8 16911507 IC50 = 2600 nM T40097 CPY3G0 16912155 IC50 = 2300 nM T40097 C5IYQ1 17027307 IC50 = 600 nM T40097 CZN7E9 17144353 IC50 = 6000 nM T40097 CJB1G8 17144354 IC50 = 5400 nM T40097 CQ32TU 17144355 IC50 = 4300 nM T40097 C5P6JV 17173055 IC50 = 12500 nM T40097 CQJ12W 17496132 IC50 > 50000 nM T40097 CIO78T 17551446 IC50 = 83500 nM T40097 C8VG1K 17567050 IC50 = 7600 nM T40097 C1GKL6 17758020 IC50 > 40000 nM T40097 CWH37T 17758574 IC50 = 31000 nM T40097 CM3W4G 20626890 IC50 = 5930 nM T40097 COS4H1 20626909 IC50 = 650 nM T40097 C9BI2Y 23060924 IC50 = 1400 nM T40097 C2NLE3 23060985 IC50 = 860 nM T40097 CYK74S 23434550 IC50 = 2750 nM T40097 CM2UY0 23647201 IC50 = 980 nM T40097 C3UOY0 23647202 IC50 = 920 nM T40097 C40DPW 23647203 IC50 > 10000 nM T40097 CGRL48 23647204 IC50 = 5140 nM T40097 CW2I3J 23647205 IC50 > 10000 nM T40097 C0LPF5 23647206 IC50 > 10000 nM T40097 C2WHZ1 23647207 IC50 > 10000 nM T40097 CT3NW4 23647208 IC50 > 10000 nM T40097 CC6X5S 23647209 IC50 > 10000 nM T40097 CF3XS2 23647210 IC50 = 4590 nM T40097 C7HF9E 23647211 IC50 = 2780 nM T40097 CQ87FP 23647212 IC50 = 5430 nM T40097 C41SLE 23647213 IC50 > 10000 nM T40097 CLB4D9 23647214 IC50 > 10000 nM T40097 CK5LD8 23647215 IC50 > 10000 nM T40097 CNOA35 23647216 IC50 = 960 nM T40097 CQDB80 23647217 IC50 = 1310 nM T40097 C1MYT5 23647218 IC50 = 520 nM T40097 CS69RG 23647219 IC50 = 2640 nM T40097 CIDG42 23647220 IC50 > 10000 nM T40097 CJ3QI9 23647221 IC50 > 10000 nM T40097 CA26PG 23647222 IC50 > 10000 nM T40097 CKP16G 23647223 IC50 = 2410 nM T40097 C8Y1MN 23647224 IC50 > 10000 nM T40097 C0PXL4 23647225 IC50 = 2740 nM T40097 C5AHM8 23647226 IC50 = 2830 nM T40097 C0E4ZY 23647227 IC50 = 750 nM T40097 CY3L0H 23647228 IC50 = 780 nM T40097 CM10AZ 23647229 IC50 = 500 nM T40097 C29TJW 23647230 IC50 = 430 nM T40097 C4NL5H 23647231 IC50 = 4410 nM T40097 C62DWL 23647232 IC50 = 7640 nM T40097 C7C4IX 23647233 IC50 = 8770 nM T40097 C4W5GQ 23647234 IC50 = 7670 nM T40097 C8QE9S 23647235 IC50 = 4190 nM T40097 CR2V5H 23647236 IC50 = 1750 nM T40097 CGXB32 23647237 IC50 = 75 nM T40097 CBV3A2 23647238 IC50 = 1500 nM T40097 CVMZ10 23647239 IC50 = 44700 nM T40097 CN2S4C 23647242 IC50 > 100000 nM T40097 C0IS4R 23647244 IC50 = 700 nM T40097 C32VGZ 23647247 IC50 = 18200 nM T40097 C5ZM7W 23647248 IC50 = 400 nM T40097 C4W9HQ 23647249 IC50 > 100000 nM T40097 CU2P1C 23647250 IC50 = 76 nM T40097 CU02AM 23647251 IC50 = 25 nM T40097 C2ND5K 23647252 IC50 = 35 nM T40097 CN8F5Y 23647254 IC50 = 35 nM T40097 C1ZE9J 23647255 IC50 = 28 nM T40097 CD9AC7 23647256 IC50 = 29 nM T40097 CTLM13 23647257 IC50 = 157 nM T40097 C6J3VB 23647258 IC50 = 93 nM T40097 CEGH40 23647259 IC50 = 278 nM T40097 CKT0M3 23647260 IC50 = 391 nM T40097 CO2N9V 23647261 IC50 = 186 nM T40097 CK0U2E 23647262 IC50 = 33 nM T40097 C1TZ4I 23647263 IC50 = 37 nM T40097 C6H5EU 23647264 IC50 = 46 nM T40097 C1LBF6 23647265 IC50 = 55 nM T40097 C2ZQ6H 23647266 IC50 = 85 nM T40097 CKUQ73 23647267 IC50 = 705 nM T40097 CC07GV 23647268 IC50 = 204 nM T40097 CS69KN 23647269 IC50 = 82 nM T40097 C9WD6T 23647270 IC50 = 21 nM T40097 C7N6VC 23647271 IC50 = 32 nM T40097 C0QAB8 23647272 IC50 = 20 nM T40097 CVOT06 24535122 IC50 = 2000 nM T40097 CV9U8E 24745781 IC50 > 10000 nM T40097 C7YG1N 24759534 IC50 = 12000 nM T40097 C16DKC 24810995 IC50 > 10000 nM T40097 CC8Y1U 24810996 IC50 = 2900 nM T40097 CH21WG 24810997 IC50 = 840 nM T40097 CQ1D8M 24810999 IC50 = 3600 nM T40097 CNI4W8 24811099 IC50 = 6300 nM T40097 C0MXK3 24811100 IC50 = 1800 nM T40097 CFZN51 24811101 IC50 = 800 nM T40097 CRF71M 24811102 IC50 = 580 nM T40097 CB8A2T 24811103 IC50 > 10000 nM T40097 CCP2M3 24822704 IC50 > 50000 nM T40097 CJ7M8K 24823663 IC50 = 24 nM T40097 CLP68C 24823665 IC50 = 29 nM T40097 CRV5C7 24823814 IC50 = 39 nM T40097 CSW3D9 24823964 IC50 = 63 nM T40097 CL61YV 24824104 IC50 = 74 nM T40097 CX0S9L 24854902 IC50 > 10000 nM T40097 C1SVT2 24854903 IC50 > 10000 nM T40097 C4OWF8 24875373 IC50 = 74 nM T40097 C3V1PU 24881467 IC50 = 20 nM T40097 C13QYB 24884503 IC50 > 2000 nM T40097 CY8L7E 24896769 IC50 > 10000 nM T40097 C8DG1Y 24941253 IC50 > 10000 nM T40097 C42HGN 24957306 IC50 = 55 nM T40097 CK4W5P 24957308 IC50 = 65 nM T40097 CE8KJ9 24960632 IC50 = 140 nM T40097 C9WOQ0 24960635 IC50 = 250 nM T40097 C6B0IM 24961360 IC50 = 23 nM T40097 CU7I2E 24963046 IC50 > 10000 nM T40097 CD0TB3 25024184 IC50 = 166 nM T40097 C4OA5D 25113170 IC50 = 13 nM T40097 CM2K9V 25119432 IC50 = 80 nM T40097 CF7C5B 25129829 IC50 > 10000 nM T40097 CXNM84 25129830 IC50 > 10000 nM T40097 CY2S1P 25129831 IC50 > 10000 nM T40097 C9ZKH4 25174103 IC50 = 73 nM T40097 CYTV68 25181985 IC50 = 18 nM T40097 C5KIE7 25182113 IC50 = 30 nM T40097 C6FGQ1 25206346 IC50 > 10000 nM T40097 CEFT59 25210489 IC50 = 240 nM T40097 CEU0R6 25211574 IC50 = 1995 nM T40097 C3SYO4 25211575 IC50 = 1585 nM T40097 CG40OH 25211676 IC50 = 3162 nM T40097 CXE16F 25218564 IC50 = 3162 nM T40097 C3RH2Q 25218565 IC50 = 3891 nM T40097 C20THL 25218566 IC50 = 631 nM T40097 C25DJY 25218567 IC50 = 1258 nM T40097 CHM29R 25218568 IC50 = 5011 nM T40097 CI78TL 25218569 IC50 = 501 nM T40097 CG29EY 25218570 IC50 = 1258 nM T40097 C16ISR 25218571 IC50 = 3981 nM T40097 C9FAL8 25218572 IC50 = 10000 nM T40097 C9G2ZM 25218573 IC50 = 10000 nM T40097 CB03GW 25218574 IC50 = 126 nM T40097 CC39RK 25218575 IC50 = 1000 nM T40097 C0ZJ3O 25218576 IC50 = 1995 nM T40097 CRM7N5 25218577 IC50 = 3162 nM T40097 CR3KE8 25218578 IC50 = 794 nM T40097 C6T9AO 25218579 IC50 = 1000 nM T40097 CGK1O0 25218580 IC50 = 1259 nM T40097 C0S4UP 25218581 IC50 = 1995 nM T40097 C89DVN 25218582 IC50 = 631 nM T40097 CLM18I 25218583 IC50 = 126 nM T40097 CBSY10 25218584 IC50 = 1585 nM T40097 CDYZ78 25218585 IC50 = 794 nM T40097 CCL2O3 25218586 IC50 = 251 nM T40097 CR3UY7 25218587 IC50 = 1585 nM T40097 CN5X1G 25218588 IC50 = 100 nM T40097 C04PGY 25218589 IC50 = 7943 nM T40097 CD7KC4 25218590 IC50 = 6310 nM T40097 C1ODR5 25218591 IC50 = 2512 nM T40097 CYB58C 25218592 IC50 = 7943 nM T40097 CO0RF6 25218593 IC50 = 12 nM T40097 CMF51N 25222038 IC50 = 99 nM T40097 C15DIA 25222587 IC50 = 39 nM T40097 CV7AG6 25660569 IC50 = 400 nM T40097 C0NR9F 26644345 IC50 = 3981.07 nM T40097 C5GZ8L 26704995 IC50 = 600 nM T40097 CU1M8N 33657234 IC50 = 100 nM T40097 CD2OC8 34676239 IC50 = 6309.57 nM T40097 C75GBV 40805001 IC50 = 3200 nM T40097 C1AFJ7 41107918 IC50 = 1800 nM T40097 CTV2G9 41362568 IC50 > 25000 nM T40097 CRY5L4 42537838 IC50 = 360 nM T40097 CU9E4P 42629114 IC50 > 10000 nM T40097 CI5AE0 43623574 IC50 = 6600 nM T40097 C0HB4C 44129168 IC50 = 14100 nM T40097 CX16AN 44138038 Ki = 9 nM T40097 CO42DC 44138048 IC50 = 100000 nM T40097 CL65QV 44138049 IC50 > 100000 nM T40097 CPT6F0 44224261 IC50 = 140 nM T40097 CEL61X 44229839 IC50 > 10000 nM T40097 CMRG01 44236943 IC50 = 4100 nM T40097 C0HM6Z 44236944 IC50 = 630 nM T40097 CRT04D 44236945 IC50 = 1500 nM T40097 C46EDI 44236946 IC50 = 400 nM T40097 C37IRD 44236947 IC50 = 180 nM T40097 CGSA21 44236948 IC50 = 270 nM T40097 CGO6L3 44236949 IC50 = 880 nM T40097 CYV31G 44236950 IC50 = 900 nM T40097 C2D4LE 44236951 IC50 = 1200 nM T40097 C6IGK2 44236952 IC50 > 20000 nM T40097 CFU45N 44236953 IC50 = 6300 nM T40097 C07YUQ 44236954 IC50 = 180 nM T40097 C8HPQ7 44236955 IC50 = 110 nM T40097 CG8KU3 44236956 IC50 > 20000 nM T40097 CLK0U1 44236957 IC50 > 20000 nM T40097 C9L3XK 44236958 IC50 > 20000 nM T40097 CRJ9F0 44236959 IC50 > 20000 nM T40097 CBXL42 44236960 IC50 = 330 nM T40097 C9HR2S 44236961 IC50 = 1800 nM T40097 CW3PO4 44236964 IC50 = 4500 nM T40097 C82AFZ 44236967 IC50 = 1800 nM T40097 CTH0D7 44236968 IC50 = 7100 nM T40097 COF30J 44236969 IC50 > 20000 nM T40097 C6J0UF 44236970 IC50 > 20000 nM T40097 CP81MF 44236971 IC50 = 90 nM T40097 CTHS64 44236972 IC50 = 40 nM T40097 CNL6H4 44236973 IC50 = 210 nM T40097 C87WNK 44236974 IC50 = 230 nM T40097 CJ9VI7 44236975 IC50 = 330 nM T40097 C0FT5H 44236976 IC50 = 260 nM T40097 C1HX8I 44236977 IC50 = 1400 nM T40097 CET82Q 44236978 IC50 = 110 nM T40097 C59YJV 44236979 IC50 = 3200 nM T40097 CSI8C1 44236980 IC50 = 450 nM T40097 CF2YU6 44236981 IC50 = 5800 nM T40097 C19NBZ 44236982 IC50 > 20000 nM T40097 C0KD4U 44346053 IC50 = 150 nM T40097 CZ1Y5U 44397446 IC50 = 1584.89 nM T40097 CT9I6Z 44397450 IC50 = 1584.89 nM T40097 CUQ7O6 44397681 IC50 = 5011.87 nM T40097 C7NYI2 44397684 IC50 = 3981.07 nM T40097 C8QZ5E 44397760 IC50 = 794.33 nM T40097 CR8I3D 44397783 IC50 = 1258.93 nM T40097 C2MT9X 44404797 IC50 = 81 nM T40097 CAC7Q5 44404813 IC50 = 71 nM T40097 C7F6KQ 44408641 IC50 = 122 nM T40097 C27KEP 44408669 IC50 = 219 nM T40097 CFY5E9 44408670 IC50 = 152 nM T40097 CI76KB 44408825 IC50 = 82 nM T40097 CBC3X6 44408908 IC50 = 74 nM T40097 CY8LJ5 44408909 IC50 = 125 nM T40097 C3O7GC 44408936 IC50 = 85 nM T40097 CCW09A 44408944 IC50 = 48 nM T40097 CY6EW5 44419110 IC50 = 349.95 nM T40097 CM31PI 44419111 IC50 > 10000 nM T40097 CG90BS 44419115 IC50 = 3427.68 nM T40097 CP05HO 44419116 IC50 = 1088.93 nM T40097 C9IWT5 44419118 IC50 = 2238.72 nM T40097 CNJ5F1 44419119 IC50 = 1548.82 nM T40097 CWC0G6 44419127 IC50 = 5248.07 nM T40097 CAYL35 44419128 IC50 = 1180 nM T40097 COC4P2 44419129 IC50 = 260 nM T40097 C5ZMS7 44419130 IC50 = 92.9 nM T40097 CH8WZ7 44419135 IC50 = 199.99 nM T40097 CRI6V9 44419136 IC50 = 429.54 nM T40097 CY6DK0 44419137 IC50 = 66 nM T40097 CZP46I 44419138 IC50 = 59 nM T40097 CQT30U 44419143 IC50 = 42.95 nM T40097 C8J6MZ 44419144 IC50 = 81 nM T40097 CYM3X7 44419145 IC50 = 53.95 nM T40097 CHG96R 44419146 IC50 = 92.9 nM T40097 CLX1B5 44419150 IC50 = 269.77 nM T40097 C0CLT1 44419151 IC50 = 250.03 nM T40097 CKL2A8 44419152 IC50 = 120 nM T40097 C9ED6R 44419153 IC50 = 1599.56 nM T40097 CJ1RE0 44419155 IC50 = 570.16 nM T40097 C65XAW 44419156 IC50 = 1990 nM T40097 CQW93F 44419157 IC50 = 7294.58 nM T40097 CMCF90 44419158 IC50 = 179.89 nM T40097 C40QDE 44419161 IC50 = 319.89 nM T40097 C3JW9E 44419162 IC50 = 529.66 nM T40097 CNX3P1 44419163 IC50 = 180 nM T40097 C3GV8D 44419164 IC50 = 1500 nM T40097 C1XI7E 44419168 IC50 = 620 nM T40097 CDIL57 44419169 IC50 = 47.97 nM T40097 C4YQD8 44419170 IC50 = 76.03 nM T40097 CQE6D3 44419174 IC50 = 150 nM T40097 C76JCA 44419175 IC50 = 1448.77 nM T40097 CK4Z6B 44419182 IC50 = 169.82 nM T40097 CST57V 44419183 IC50 = 300 nM T40097 CR9ON4 44419190 IC50 = 1640 nM T40097 C1RL3U 44419191 IC50 = 429.54 nM T40097 C8IJ2U 44419202 IC50 = 87.9 nM T40097 C5KBX0 44419203 IC50 = 389.94 nM T40097 CRGD85 44419210 IC50 = 419.76 nM T40097 CP1C8D 44419211 IC50 = 66.99 nM T40097 CO9AK1 44419214 IC50 = 1180 nM T40097 CE20PN 44419215 IC50 = 2432.2 nM T40097 C4V6YN 44419216 IC50 = 32 nM T40097 CF4I1R 44419217 IC50 = 85 nM T40097 C13EQD 44419220 IC50 = 2930 nM T40097 C1KQL5 44419221 IC50 = 410 nM T40097 CD8EB4 44419222 IC50 = 95.94 nM T40097 CCBL15 44419223 IC50 = 820 nM T40097 CY1Q7N 44419226 IC50 = 79 nM T40097 CXR83C 44419227 IC50 = 317.69 nM T40097 CO91FC 44431824 IC50 > 10000 nM T40097 C2C4SX 44431829 IC50 > 10000 nM T40097 C9Y1ID 44431830 IC50 > 10000 nM T40097 CU20ER 44431831 IC50 > 10000 nM T40097 CL87AX 44431832 IC50 > 10000 nM T40097 CA61VJ 44431833 IC50 > 10000 nM T40097 C1KW0V 44431834 IC50 > 10000 nM T40097 C2NS4X 44439209 IC50 > 10000 nM T40097 C1LHZ9 44439211 IC50 = 6400 nM T40097 CUZH09 44439213 IC50 = 30 nM T40097 C9B1UC 44439214 IC50 = 61 nM T40097 CCR0I2 44439215 IC50 = 50 nM T40097 C58GAX 44439216 IC50 = 130 nM T40097 CAX8F5 44440161 IC50 = 92 nM T40097 CK9H1G 44440214 IC50 = 74 nM T40097 CDF70Q 44440215 IC50 = 41 nM T40097 CK8L4U 44440216 IC50 = 457 nM T40097 CM2E3N 44440217 IC50 = 59 nM T40097 CWL30H 44440218 IC50 = 71 nM T40097 C6RD3G 44440219 IC50 = 360 nM T40097 CIAJ70 44440220 IC50 = 1340 nM T40097 C52CDB 44440221 IC50 = 29 nM T40097 C2OC7L 44440222 IC50 = 139 nM T40097 CFZS24 44440223 IC50 = 60 nM T40097 CSA87R 44440224 IC50 = 15 nM T40097 CH76CV 44440225 IC50 = 13 nM T40097 CP80UK 44440226 IC50 = 15 nM T40097 CFI06W 44440227 IC50 = 18 nM T40097 CKSO82 44440228 IC50 = 67 nM T40097 C8HWI1 44440229 IC50 = 57 nM T40097 CVD97U 44440230 IC50 = 15 nM T40097 C1B0TO 44440234 IC50 = 47 nM T40097 CS5PY4 44440235 IC50 = 520 nM T40097 C9AV4C 44440236 IC50 = 22 nM T40097 C0SQE3 44449102 IC50 = 3801 nM T40097 C07MAX 44451531 IC50 = 3.3 nM T40097 CN48AD 44451535 IC50 = 7.6 nM T40097 CRJ2G5 44451555 IC50 = 48 nM T40097 CNIQ82 44451560 IC50 = 10 nM T40097 C5X6YO 44451561 IC50 = 10 nM T40097 C87NZM 44451562 IC50 = 10 nM T40097 C18SFJ 44451585 IC50 = 12 nM T40097 C5Z4HI 44451588 IC50 = 11 nM T40097 C73OWC 44451589 IC50 = 11 nM T40097 CBZ79T 44451607 IC50 = 43 nM T40097 CL8YP9 44451612 IC50 = 9.4 nM T40097 C4KDY6 44451615 IC50 = 33 nM T40097 C3POR4 44451616 IC50 = 7.3 nM T40097 CK6YR8 44451635 IC50 = 14 nM T40097 CT3F7S 44451638 IC50 = 89 nM T40097 C07NVI 44451642 IC50 = 43 nM T40097 CNQ49Y 44451663 IC50 = 42 nM T40097 C6UA5O 44451666 IC50 = 79 nM T40097 C9MRD0 44451669 IC50 = 8.6 nM T40097 CEC1L4 44451670 IC50 = 6.8 nM T40097 CEPG82 44451685 IC50 = 100 nM T40097 CH0CT1 44451687 IC50 = 1100 nM T40097 C5MQX7 44451688 IC50 = 190 nM T40097 C8K5LD 44451690 IC50 = 86 nM T40097 CLY8P9 44451693 IC50 = 28 nM T40097 C0HY3S 44451713 IC50 = 450 nM T40097 CZM16V 44451763 IC50 = 63 nM T40097 C4MU2Z 44451764 IC50 = 21 nM T40097 CW3JI7 44451791 IC50 = 28 nM T40097 CSFX51 44451793 IC50 = 59 nM T40097 C4T6VG 44451795 IC50 = 8800 nM T40097 CCD6Z7 44451820 IC50 = 140 nM T40097 CI2OX1 44451850 IC50 = 1500 nM T40097 CSY06K 44451882 IC50 = 61 nM T40097 CW5X1P 44451905 IC50 = 95 nM T40097 C8DEF1 44517631 IC50 = 4220 nM T40097 CU80BP 44517743 IC50 > 10000 nM T40097 CYH6P3 44520205 IC50 > 10000 nM T40097 C3VRO9 44557921 IC50 > 10000 nM T40097 CF90OX 44576212 IC50 = 175000 nM T40097 CWQ61M 44576547 IC50 = 1499.68 nM T40097 C3Y4OS 44576549 IC50 = 1640.59 nM T40097 CEP8R1 44585572 IC50 = 1200 nM T40097 CLA8O9 44585590 IC50 = 1400 nM T40097 C6K5CT 44585591 IC50 = 4500 nM T40097 CC5W9J 44586319 IC50 = 2080 nM T40097 CMKH90 44591675 Ki = 48 nM T40097 C2X7DJ 44591676 Ki = 151 nM T40097 CUL5A2 44591677 Ki = 27 nM T40097 C2SP5J 44591702 Ki = 315 nM T40097 C2S4PZ 44591703 Ki = 26 nM T40097 C7GL4H 44591704 Ki = 1570 nM T40097 CLKG07 44591705 Ki = 2730 nM T40097 COZ16T 44591706 Ki = 381 nM T40097 CHD64X 44591707 Ki = 43 nM T40097 C8T1LV 44591735 Ki = 169 nM T40097 CB1AF0 44591736 Ki = 530 nM T40097 CV26OD 44591737 Ki = 101 nM T40097 CY26UI 44591738 Ki = 162 nM T40097 C3D8RZ 44591739 Ki = 12 nM T40097 C5Z3LI 44591740 Ki = 12 nM T40097 C6OZB5 44591767 Ki = 36 nM T40097 CU23PY 44591768 Ki = 9 nM T40097 COHK45 44591769 Ki = 28 nM T40097 CV8F0R 44593854 IC50 > 10000 nM T40097 CZ8XI5 44627578 IC50 = 535 nM T40097 CN30CM 44627580 IC50 = 123 nM T40097 C7NU3G 44627581 IC50 = 19 nM T40097 CDF41Q 44627582 IC50 = 16 nM T40097 CKI17J 44627583 IC50 = 113 nM T40097 C7EK0M 44627681 IC50 = 54 nM T40097 C8RVP9 44627682 IC50 = 45 nM T40097 C6E2LI 44627683 IC50 = 97 nM T40097 C21IGV 44627684 IC50 = 102 nM T40097 CJ0LU4 45104966 IC50 = 283 nM T40097 CJ32SA 45203151 IC50 >= 20000 nM T40097 C2JVA4 45270368 IC50 = 79 nM T40097 C6E2SC 45482700 IC50 > 10000 nM T40097 CZXH74 45482750 IC50 > 10000 nM T40097 CUA97D 46209401 IC50 > 10000 nM T40097 CZ58FY 46215814 IC50 > 10000 nM T40097 CY3HW5 46224684 IC50 = 520 nM T40097 C6M7CK 46232266 IC50 = 10000 nM T40097 CJZA45 46232267 IC50 = 6700 nM T40097 C6EX9F 46232268 IC50 = 9100 nM T40097 C3PLE6 46232269 IC50 = 4800 nM T40097 C3U8HV 46232270 IC50 = 5700 nM T40097 CYA73D 46232312 IC50 = 3000 nM T40097 C9JDL8 46232313 IC50 = 100000 nM T40097 CW2G7D 46868853 IC50 = 11 nM T40097 CR57OZ 46868855 IC50 = 226 nM T40097 CI8YE5 46868856 IC50 = 12 nM T40097 C94EPL 46868925 IC50 = 3 nM T40097 C0GU4D 46868930 IC50 = 140 nM T40097 C9ULP0 46869071 IC50 = 3200 nM T40097 CU52JS 46869075 IC50 = 3200 nM T40097 CFQT10 46869147 IC50 = 24100 nM T40097 CEK2I5 46869149 IC50 = 710 nM T40097 C2XQ4K 46869223 IC50 = 3400 nM T40097 C8U1AH 46869285 IC50 = 5 nM T40097 CKTD23 46869290 IC50 = 81 nM T40097 CV57OI 46869490 IC50 = 7 nM T40097 C9XHK0 46869491 IC50 = 8 nM T40097 C47JSD 46869493 IC50 = 3 nM T40097 C65NDB 46869609 IC50 = 30300 nM T40097 CP2A4Y 46869611 IC50 = 250 nM T40097 CQ0AU8 46869671 IC50 = 43600 nM T40097 C4RS7M 46869672 IC50 = 331 nM T40097 C1VZM6 46869673 IC50 = 4 nM T40097 CYI69K 46869674 IC50 = 15 nM T40097 C2PC6T 46869677 IC50 = 830 nM T40097 CSL2N6 46869740 IC50 = 3400 nM T40097 C6V9CD 46869741 IC50 = 32 nM T40097 CZCQ05 46869742 IC50 = 790 nM T40097 C09GAW 46869745 IC50 = 105 nM T40097 CVBG98 46869815 IC50 = 298 nM T40097 CU2D5N 46869816 IC50 = 15 nM T40097 C8WH7Q 46869817 IC50 = 45 nM T40097 CFOX43 46869876 IC50 = 463 nM T40097 CE0CY1 46869877 IC50 = 270 nM T40097 C2DW6T 46869878 IC50 = 28 nM T40097 C19DQG 46869879 IC50 = 42 nM T40097 CR1OH0 46869880 IC50 = 9 nM T40097 C8SFI1 46869881 IC50 = 6 nM T40097 CD1YH9 46869882 IC50 = 25 nM T40097 CLS29B 46872626 IC50 > 10000 nM T40097 CRKV43 46884199 Ki = 3 nM T40097 CGX79T 46896670 IC50 = 87 nM T40097 CA8M5I 46926712 IC50 = 2700 nM T40097 C94ZXN 46926787 IC50 > 25000 nM T40097 CHSF07 49806372 IC50 > 1000 nM T40097 CBS64G 49830252 IC50 = 92000 nM T40097 CS18HZ 49839481 IC50 = 48 nM T40097 CDR47S 49867175 IC50 = 400 nM T40097 CH4FY5 50941455 IC50 = 1000 nM T40097 CBR71Y 50941538 IC50 = 420 nM T40097 C4BN7W 50941539 IC50 = 700 nM T40097 CHIY40 50943203 IC50 = 6 nM T40097 CEOB58 50943512 IC50 = 29 nM T40097 CGZC83 50943588 IC50 = 3 nM T40097 CEX3H8 50943666 IC50 = 5 nM T40097 C1JY2U 50943668 IC50 = 10 nM T40097 CPS4I5 50943669 IC50 = 3 nM T40097 C83EZX 50943670 IC50 = 7 nM T40097 CNUZ80 50943753 IC50 = 12 nM T40097 COU4W2 50943754 IC50 = 8 nM T40097 C2J7ZP 50943755 IC50 = 7 nM T40097 C5GPU9 51346941 IC50 = 50 nM T40097 CEQN27 52936621 Ki > 1000 nM T40097 CM24LF 52938983 IC50 = 1592 nM T40097 CA7HQ9 52941011 IC50 = 300 nM T40097 CA6BH5 52941226 IC50 = 2100 nM T40097 CMXC68 52941286 IC50 = 1100 nM T40097 C0DSA8 52941649 IC50 = 6300 nM T40097 C3BKR7 52942436 IC50 = 6400 nM T40097 C8R9SA 52942482 IC50 > 50000 nM T40097 CAC3J5 52942507 IC50 = 1400 nM T40097 CTPH98 52942532 IC50 > 50000 nM T40097 CS8VA0 52943431 IC50 = 2600 nM T40097 CJU79I 52943626 IC50 = 890 nM T40097 C07JYV 52944873 IC50 = 1800 nM T40097 CB1UJ7 52944909 IC50 = 1700 nM T40097 CD2WZ5 52944914 IC50 = 1000 nM T40097 CY9B7D 52944962 IC50 > 50000 nM T40097 C1Z7KR 52946059 IC50 = 26900 nM T40097 CCMX82 52946092 IC50 = 23400 nM T40097 CPIK13 52946145 IC50 = 7000 nM T40097 C67TBV 52946152 IC50 = 500 nM T40097 C6OH8X 52946172 IC50 > 50000 nM T40097 CC6Z1J 52947386 IC50 = 2300 nM T40097 CC5P4R 52947399 IC50 > 50000 nM T40097 C9O7FN 52947421 IC50 > 50000 nM T40097 C72TPI 52947422 IC50 > 50000 nM T40097 C3R4FI 52948519 IC50 = 530 nM T40097 CLU92X 52948565 IC50 = 23900 nM T40097 CDXL70 52948593 IC50 = 410 nM T40097 CMT75N 52949817 IC50 = 270 nM T40097 CBAD62 52949818 IC50 = 300 nM T40097 CSOB70 52950113 IC50 = 460 nM T40097 CW2KE5 53317337 IC50 = 18900 nM T40097 CJQN83 53317338 IC50 = 1050 nM T40097 CJ2P3V 53317339 IC50 = 597 nM T40097 C9E3FV 53317340 IC50 = 284 nM T40097 CBTX53 53317412 IC50 > 50000 nM T40097 COCN94 53317413 IC50 = 2200 nM T40097 CHC29T 53317414 IC50 > 50000 nM T40097 C82LCE 53317415 IC50 > 50000 nM T40097 CR0DJ1 53317416 IC50 = 3800 nM T40097 C28JAP 53317417 IC50 = 900 nM T40097 C8Q0OR 53318506 IC50 = 31 nM T40097 CP7T3N 53318709 IC50 > 500 nM T40097 CKD47I 53319944 IC50 = 295 nM T40097 CP7BR1 53319945 IC50 = 686 nM T40097 C3TAC2 53320021 IC50 > 5000 nM T40097 COPI53 53321333 IC50 = 7200 nM T40097 C0GLS5 53321334 IC50 = 4600 nM T40097 C2V0QU 53321577 IC50 = 3300 nM T40097 CG8KC9 53322569 IC50 = 19300 nM T40097 C3SA1K 53322570 IC50 = 350 nM T40097 COG9J2 53322644 IC50 > 50000 nM T40097 CUR1A6 53322645 IC50 = 740 nM T40097 C25OEY 53322984 IC50 = 78 nM T40097 CK8Y5F 53323911 IC50 = 95 nM T40097 C9SHJ0 53323985 IC50 = 1800 nM T40097 C49MDG 53323986 IC50 = 1800 nM T40097 C3AVG0 53323987 IC50 = 4200 nM T40097 C18SCR 53323988 IC50 = 110 nM T40097 C38RXW 53323989 IC50 = 420 nM T40097 CXWB94 53325188 IC50 = 55 nM T40097 C8VPW5 53325283 IC50 = 990 nM T40097 CA3X2Q 53325284 IC50 = 3900 nM T40097 CIG7X9 53325285 IC50 = 2600 nM T40097 C4A8JK 53325286 IC50 = 1400 nM T40097 CI1RT4 53325287 IC50 > 5000 nM T40097 CNT50E 53325288 IC50 = 360 nM T40097 CR91NJ 53325555 IC50 = 590 nM T40097 CBW0G7 53326484 IC50 = 15580 nM T40097 CV7I4O 53326555 IC50 = 740 nM T40097 C27IBZ 53326556 IC50 = 5700 nM T40097 C5UK3J 53326557 IC50 = 1700 nM T40097 CVJ6K9 53326558 IC50 = 4500 nM T40097 C8NA4L 53384644 IC50 > 30000 nM T40097 CD0ZI6 53469858 IC50 = 7150 nM T40097 CY8RB7 54580142 IC50 > 100000 nM T40097 C1ETG7 54580171 IC50 > 25000 nM T40097 C67UCX 54580172 IC50 = 1800 nM T40097 CXLV70 54580173 IC50 = 9700 nM T40097 C1PJX9 54581164 IC50 > 25000 nM T40097 CA5HJ1 54581165 IC50 = 10200 nM T40097 CMFO90 54581166 IC50 = 1900 nM T40097 CB4TJ8 54581287 IC50 = 40 nM T40097 CT3JS6 54581291 IC50 = 30 nM T40097 CEP18Y 54581359 IC50 > 50000 nM T40097 C6JPE1 54581360 IC50 > 50000 nM T40097 CD2YU5 54581361 IC50 > 50000 nM T40097 C49RNQ 54581362 IC50 > 50000 nM T40097 CA8U3P 54581363 IC50 > 50000 nM T40097 C5V6OY 54582175 IC50 = 19730 nM T40097 COK26W 54582187 IC50 > 25000 nM T40097 CF4SZ1 54582188 IC50 = 8300 nM T40097 CSMB26 54582189 IC50 = 8100 nM T40097 CAO0L7 54582190 IC50 = 2500 nM T40097 CBTV46 54582191 IC50 = 2500 nM T40097 CT2UJ1 54583154 IC50 > 25000 nM T40097 CNEF71 54583155 IC50 = 2900 nM T40097 C8WSJ9 54583156 IC50 > 25000 nM T40097 CY18TP 54583157 IC50 = 7600 nM T40097 CQ85PS 54583158 IC50 = 4900 nM T40097 C1OM6E 54583278 IC50 = 10 nM T40097 CCO5I2 54583368 IC50 > 50000 nM T40097 CECO89 54583369 IC50 > 50000 nM T40097 C2OSA7 54584118 IC50 > 25000 nM T40097 CQXD91 54584145 IC50 = 6400 nM T40097 CZ9OC1 54584146 IC50 = 5800 nM T40097 C7H9XW 54584147 IC50 = 20900 nM T40097 CA0NT4 54584148 IC50 = 3400 nM T40097 CO48MC 54584149 IC50 = 8200 nM T40097 CYF0K8 54584150 IC50 = 7400 nM T40097 C10NCB 54584151 IC50 = 3100 nM T40097 CM1TU0 54584242 IC50 = 90 nM T40097 CP6K3I 54584243 IC50 = 50 nM T40097 CRKI30 54584315 IC50 > 50000 nM T40097 C3P2HM 54584316 IC50 > 50000 nM T40097 CL69AG 54584317 IC50 = 6850 nM T40097 C9BYF3 54585051 IC50 > 25000 nM T40097 C8ZU7H 54585083 IC50 > 100000 nM T40097 CUZP45 54585084 IC50 = 1800 nM T40097 CI1M7Q 54585085 IC50 = 5800 nM T40097 CY7V9F 54585117 IC50 = 9400 nM T40097 CT16HO 54585212 IC50 = 20 nM T40097 CC8YN2 54585285 IC50 > 50000 nM T40097 CGA8X9 54585286 IC50 > 50000 nM T40097 CV69FU 54585287 IC50 > 50000 nM T40097 CR1X8Y 54585288 IC50 = 24300 nM T40097 CTY84H 54585289 IC50 > 50000 nM T40097 CWE79L 54585290 IC50 > 50000 nM T40097 C0FAG2 54585291 IC50 = 41900 nM T40097 CNLU49 54585292 IC50 > 50000 nM T40097 CNUP53 54586040 IC50 = 480 nM T40097 CJ76FS 54586056 IC50 > 25000 nM T40097 CU1KO5 54586057 IC50 > 25000 nM T40097 CK8L6V 54586058 IC50 = 2600 nM T40097 CUD8J0 54586233 IC50 > 50000 nM T40097 CU4F9E 54587045 IC50 > 50000 nM T40097 CH92LK 54587046 IC50 = 3400 nM T40097 C9T4OD 54587047 IC50 = 3600 nM T40097 C4JN0R 54587048 IC50 = 2500 nM T40097 C1V8HM 54587177 IC50 = 100 nM T40097 CO1JB2 54587178 IC50 = 10 nM T40097 CA5N6I 54587258 IC50 > 50000 nM T40097 CKX15Q 54587259 IC50 > 50000 nM T40097 CKQS27 54587260 IC50 > 50000 nM T40097 C57LBW 54587261 IC50 > 50000 nM T40097 CFRA47 54675539 IC50 = 37 nM T40097 CG4WB5 54675542 IC50 = 118 nM T40097 C1QYV4 54675574 IC50 = 93.7 nM T40097 C0I4FV 54764508 IC50 = 27 nM T40097 C18TKF 54764593 IC50 = 4 nM T40097 CN9QD7 56643097 IC50 > 10000 nM T40097 CG78UW 56658171 IC50 = 10 nM T40097 C31LBA 56658172 IC50 = 14000 nM T40097 CNB94K 56658173 IC50 = 0.9 nM T40097 C7LDZ3 56658303 IC50 = 178 nM T40097 C0MW6D 56658304 IC50 = 8 nM T40097 CK18JP 56661802 IC50 = 14 nM T40097 CE1O3B 56661803 IC50 = 9 nM T40097 CSJ6A9 56665092 IC50 = 1 nM T40097 C7HA6J 56665093 IC50 = 2 nM T40097 CS5HP6 56665245 IC50 = 17 nM T40097 C4SO3M 56665246 IC50 = 4 nM T40097 CE2PY0 56665247 IC50 = 2 nM T40097 C9AW1E 56668539 IC50 = 13 nM T40097 C0MR6D 56668696 IC50 = 4 nM T40097 CXF3R9 56668697 IC50 = 11 nM T40097 CDKS47 56671909 IC50 < 500 nM T40097 CU3I2J 56672173 IC50 = 31 nM T40097 CJ9I6K 56672174 IC50 = 1 nM T40097 CD5NZ4 56672175 IC50 = 7 nM T40097 CRAK61 56675421 IC50 = 4 nM T40097 CG3ZU0 56678888 IC50 = 21 nM T40097 CAP1M2 56682209 IC50 = 16 nM T40097 C9DO8G 56682210 IC50 = 1 nM T40097 CTO6N5 56834943 IC50 = 270 nM T40097 CU5D8R 57339131 IC50 = 190 nM T40097 C97SLT 57340680 IC50 = 809 nM T40097 C0UDN5 57340685 IC50 = 1.5 nM T40097 CDP45J 57390517 IC50 = 2500 nM T40097 C28LIB 57390518 IC50 = 1100 nM T40097 C8DZ1N 57390519 IC50 = 75 nM T40097 C7K4LJ 57390520 IC50 = 2600 nM T40097 C32DFY 57390767 IC50 = 100 nM T40097 C32FUN 57390769 IC50 = 53 nM T40097 CHU75J 57390951 IC50 = 1200 nM T40097 CG51FX 57392289 IC50 = 230 nM T40097 C9EJN6 57392581 IC50 = 480 nM T40097 CSYJ61 57392738 IC50 = 160 nM T40097 C2IZ3W 57392739 IC50 = 51 nM T40097 C9P1SC 57393560 IC50 = 150 nM T40097 CVH4X0 57394043 IC50 = 160 nM T40097 CN3MB5 57394305 IC50 = 740 nM T40097 C03CNR 57394466 IC50 = 120 nM T40097 CX9B4S 57394467 IC50 = 170 nM T40097 C1EYU6 57394468 IC50 = 400 nM T40097 CV9W8C 57395293 IC50 = 180 nM T40097 CQ2A1B 57395802 IC50 = 490 nM T40097 C15YOZ 57396060 IC50 = 26 nM T40097 CL4BN7 57396061 IC50 = 35 nM T40097 CW7XA9 57397040 IC50 = 91 nM T40097 C18MFO 57397857 IC50 = 35 nM T40097 CKG0P1 57397861 IC50 = 930 nM T40097 C9A7RL 57397862 IC50 = 120 nM T40097 C4V9RN 57398023 IC50 = 120 nM T40097 CZI7A2 57398024 IC50 = 63 nM T40097 C4RJ0E 57398025 IC50 = 540 nM T40097 CH1QI7 57399519 IC50 = 22 nM T40097 CA0SR3 57399520 IC50 = 100 nM T40097 C8IFD4 57399521 IC50 = 44 nM T40097 CE76QR 57399681 IC50 = 79 nM T40097 CRNJ52 57399682 IC50 = 880 nM T40097 CT5S8H 57400156 IC50 = 680 nM T40097 C06JFP 57401276 IC50 > 20000 nM T40097 CLI72R 57401441 IC50 = 390 nM T40097 CC7N3H 57401442 IC50 = 900 nM T40097 CPY13U 57401443 IC50 = 1300 nM T40097 C8FQH3 57402785 IC50 > 10000 nM T40097 C1HD8L 57402972 IC50 = 330 nM T40097 C8ZQ3A 57403022 IC50 = 310 nM T40097 CKIX12 57403023 IC50 = 8 nM T40097 C4VKU7 57403024 IC50 = 38 nM T40097 CZ5L4E 57403025 IC50 = 3200 nM T40097 CNP8C3 57403026 IC50 = 650 nM T40097 CKE0V9 57403185 IC50 = 320 nM T40097 C7I4QD 57519510 IC50 = 67 nM T40097 CY8HG6 58017084 IC50 = 16 nM T40097 C95FNX 58082451 IC50 = 0.8 nM T40097 CXJ63M 59603829 IC50 = 18000 nM T40097 CQEU96 59603842 IC50 = 78 nM T40097 C5IN0E 59718933 IC50 = 19 nM T40097 C5CO0X 59718937 IC50 = 100 nM T40097 C1XCV6 59718972 IC50 = 120 nM T40097 C20CME 59743327 IC50 = 6.2 nM T40097 C4IM1V 59743368 IC50 = 16 nM T40097 C6VYE9 59743400 IC50 = 33 nM T40097 CJE42G 59743404 IC50 = 570 nM T40097 CUW7J8 59743407 IC50 = 4 nM T40097 C8L4KY 59743442 IC50 = 24 nM T40097 CSK8O7 59743445 IC50 = 14 nM T40097 C0MO4E 59743458 IC50 = 12 nM T40097 C5UYK1 59743461 IC50 = 14 nM T40097 CWB21E 59743477 IC50 = 56 nM T40097 C5RH4P 59743505 IC50 = 4.7 nM T40097 C3KY7N 59743507 IC50 = 9.7 nM T40097 CJ2NM1 59743549 IC50 = 34 nM T40097 CY89OP 59743571 IC50 = 4 nM T40097 C3J7CS 59846155 IC50 = 370 nM T40097 C2RCA7 59846164 IC50 = 114 nM T40097 CDA46Z 59846170 IC50 = 23 nM T40097 C86QAW 59846186 IC50 = 58 nM T40097 C20GMT 59846188 IC50 = 30 nM T40097 C5OL1V 59846192 IC50 = 130 nM T40097 CTW8X2 59846211 IC50 = 65 nM T40097 C24GXO 59846214 IC50 = 82 nM T40097 CT0K1G 59846217 IC50 = 53 nM T40097 CS2D9M 59846218 EC50 = 4100 nM T40097 C4VE3Q 59846243 IC50 = 91 nM T40097 CFPS65 59846262 IC50 = 50 nM T40097 CMZU27 59846267 IC50 = 47 nM T40097 CG3WZ7 59846277 IC50 = 38 nM T40097 CO8R0G 59846284 IC50 = 14 nM T40097 C1MR8Q 60097495 IC50 > 10000 nM T40097 CI40OG 66570843 IC50 = 12 nM T40097 CVZ67M 66816803 IC50 = 30 nM T40097 CLG56W 66940332 IC50 = 12 nM T40097 C37NKO 67129970 IC50 = 2890 nM T40097 CK80LJ 67130050 IC50 = 2750 nM T40097 CV63UL 67240318 IC50 > 10000 nM T40097 CAWC35 68621678 IC50 > 1000 nM T40097 C7GRV2 68755406 IC50 = 513 nM T40097 C5DGR9 69036886 IC50 = 10000 nM T40097 C51IQP 69309404 IC50 = 770 nM T40097 CWK7B0 70682875 IC50 = 231 nM T40097 CS3VL1 70687106 IC50 > 100000 nM T40097 CQ8HE2 70690944 IC50 > 30000 nM T40097 C13FWG 70695135 IC50 > 30000 nM T40097 C0VZB2 70697173 IC50 > 30000 nM T40097 C01ZYP 70697505 IC50 = 1035 nM T40097 C2LU7I 70702008 IC50 = 17 nM T40097 CMPK41 70702010 IC50 = 2169 nM T40097 CLB62G 70816675 EC50 = 21900 nM T40097 CJ1SW3 71452229 IC50 = 2300 nM T40097 CEBO91 71452977 IC50 > 10000 nM T40097 C3RSX5 71453059 EC50 = 14000 nM T40097 CF7N8W 71454040 IC50 = 45 nM T40097 CKT60L 71455860 Ki > 3000 nM T40097 C9S4EG 71456579 EC50 = 9000 nM T40097 C46KMY 71458431 EC50 = 9900 nM T40097 CFQ56J 71458432 EC50 = 21000 nM T40097 CHQZ25 71459584 IC50 > 10000 nM T40097 CK54JE 71460285 EC50 = 3300 nM T40097 C1DM6U 71461190 IC50 = 11000 nM T40097 C2XZO0 71576779 IC50 = 43.5 nM T40097 CZ31PU 71583657 IC50 > 10000 nM T40097 CCD0W3 71602669 IC50 = 200 nM T40097 C3D1CA 71602671 IC50 = 920 nM T40097 CG1DR3 71602672 IC50 = 93 nM T40097 CQ9A6D 71602719 IC50 = 430 nM T40097 CP01YB 71602721 IC50 = 160 nM T40097 CX60NJ 71602722 IC50 = 170 nM T40097 CHU36E 71602723 IC50 = 750 nM T40097 C7MGB8 71602768 IC50 = 1380 nM T40097 C9UY4L 71602771 IC50 = 410 nM T40097 C6O2KE 71602772 IC50 = 470 nM T40097 CS4K2F 71602818 IC50 = 800 nM T40097 CY8H5Z 71602819 IC50 = 7100 nM T40097 C60VBS 71602820 IC50 = 730 nM T40097 CI09ER 71602821 IC50 = 1200 nM T40097 C2KW8Y 71602864 IC50 = 7010 nM T40097 CAM32B 71602867 IC50 = 2300 nM T40097 CDH23B 71602868 IC50 = 1300 nM T40097 CVUG79 71602911 IC50 = 1200 nM T40097 CG0LC3 71654859 IC50 = 94 nM T40097 CHGS02 71654860 IC50 = 44 nM T40097 CTL1H9 71655707 IC50 = 6.8 nM T40097 CHX9O7 71681990 IC50 = 169 nM T40097 CLK30W 71681991 IC50 = 79.5 nM T40097 C2EYU1 71682140 IC50 = 42.8 nM T40097 C9LG1S 71682141 IC50 = 150 nM T40097 CR3HA9 71682142 IC50 = 175 nM T40097 CU8BD4 71682143 IC50 = 43 nM T40097 C5OM4V 71682298 IC50 = 1030 nM T40097 CH2RN0 71682299 IC50 = 141 nM T40097 CP56ZV 71682300 IC50 = 441 nM T40097 CJ4B7I 71682457 IC50 = 12.1 nM T40097 CD3JF9 71745086 IC50 = 970 nM T40097 C8AC4Z 72163849 IC50 = 8000 nM T40097 C3EKS1 72163850 IC50 = 2400 nM T40097 CPAC89 72163851 IC50 = 1700 nM T40097 CV15CU 72163852 IC50 = 910 nM T40097 CIO3L8 72163958 IC50 > 100000 nM T40097 C1MFV4 72163962 IC50 = 310 nM T40097 CV5S8A 72163963 IC50 = 1500 nM T40097 CT0J9N 72164072 IC50 = 570 nM T40097 CDZ7M8 72164073 IC50 = 4170 nM T40097 CC20OP 72164074 IC50 = 580 nM T40097 CO8XK4 72164075 IC50 = 1500 nM T40097 C3A7HK 72164076 IC50 = 680 nM T40097 CF06VW 72164077 IC50 = 490 nM T40097 CMEQ81 72164194 IC50 = 1980 nM T40097 CB7X5D 72164195 IC50 = 1700 nM T40097 CU9ZM5 72164196 IC50 = 33 nM T40097 C9ZYC7 72164197 IC50 = 4900 nM T40097 CN8W3X 72164198 IC50 = 67 nM T40097 CA0EZ1 72164313 IC50 = 200 nM T40097 CTL8B2 72164314 IC50 = 350 nM T40097 C6L2NG 72164315 IC50 = 360 nM T40097 C3ZDE4 72164316 IC50 = 620 nM T40097 CMH4U3 72164317 IC50 = 690 nM T40097 CR6GP3 72164438 IC50 = 270 nM T40097 CQC51G 72164439 IC50 = 59 nM T40097 CT2N9J 72164440 IC50 = 92 nM T40097 CSU3Z6 72164441 IC50 = 77 nM T40097 CECS79 72164442 IC50 = 180 nM T40097 CJKE06 72164559 IC50 = 1220 nM T40097 C5PD6V 72164560 IC50 = 430 nM T40097 CUSF60 72164561 IC50 = 250 nM T40097 CI8CA4 72164562 IC50 = 140 nM T40097 CZ4BX1 72547959 IC50 = 129 nM T40097 C9GUI2 72700745 IC50 = 41 nM T40097 CFSI04 72700746 IC50 = 47 nM T40097 C8THP4 72946274 IC50 = 160 nM T40097 CWG15I 72946453 IC50 = 152 nM T40097 C98FIU 72946656 IC50 = 33 nM T40097 CJA75F 72946661 IC50 > 20000 nM T40097 C78GOJ 72946854 IC50 = 13 nM T40097 CO61VP 72946855 IC50 = 98 nM T40097 CG4YH2 72946856 IC50 = 27 nM T40097 C0HQ6V 72947058 IC50 = 469 nM T40097 CE2Y0X 73386882 IC50 = 110 nM T40097 CJ2T9E 76332983 IC50 > 10000 nM T40097 C54KDR 86763302 IC50 > 10000 nM T40097 C4HKT5 87057579 IC50 = 2740 nM T40097 C1HW4B 89735655 IC50 = 1300 nM T40097 CQ2OB9 90292687 IC50 > 10000 nM T40097 CHI39S 90292823 IC50 > 10000 nM T40097 C0M3VU 90667135 IC50 = 1 nM T40097 C7P8TV 90667137 IC50 = 3 nM T40097 C49JZU 90667145 IC50 = 0.24 nM T40097 C7V8BN 91754589 IC50 = 7 nM T40097 CQ2G3S 91754590 IC50 = 21 nM T40097 CJQ5N6 91936970 IC50 = 1040 nM T40097 C2GNI5 101891709 IC50 = 528 nM T40097 C5DLO7 118143962 IC50 = 170 nM T40097 CK7O6G 118144051 IC50 = 3691 nM T40097 CQ29IK 118144281 IC50 = 2057 nM T40097 CZG4U9 118144359 IC50 = 537 nM T40097 C61FOL 118144367 IC50 = 5046 nM T40097 C8GU6M 118146727 IC50 = 2689 nM T40097 CY82JT 118146747 IC50 = 23 nM T40097 CIDU81 118146748 IC50 = 4544 nM T40097 C1OIF0 118146749 IC50 = 2000 nM T40097 C8TLS2 118146764 IC50 = 303 nM T40097 C32HVY 118146772 IC50 = 660 nM T40097 CULV52 118146793 IC50 = 180 nM T40097 C1MI6J 118146804 IC50 = 1226 nM T40097 CERD34 118146805 IC50 = 758 nM T40097 C48AZY 118146813 IC50 = 4728 nM T40097 CKT2Q3 118146814 IC50 = 400 nM T40097 CJ4Z3K 118146817 IC50 = 1988 nM T40097 C7Q6RW 118146819 IC50 = 400 nM T40097 CH0I3M 118146826 IC50 = 3162 nM T40097 CT29IZ 118146828 IC50 = 2625 nM T40097 CHWP46 118146849 IC50 = 1607 nM T40097 C4P9AK 118146855 IC50 = 2369 nM T40097 CT8K0N 118146868 IC50 = 1600 nM T40097 CET9N4 118146870 IC50 = 48 nM T40097 C4PBE7 118146871 IC50 = 85 nM T40097 C6LEU5 118146872 IC50 = 36 nM T40097 CX08HF 118146873 IC50 = 5385 nM T40097 CD8L5Y 118146874 IC50 = 1284 nM T40097 CNI34V 118146882 IC50 = 679 nM T40097 C8K0GC 118146884 IC50 = 7791 nM T40097 CQW3L7 118146891 IC50 = 80 nM T40097 C4O6MA 118146892 IC50 = 18 nM T40097 CZ35XB 118146932 IC50 = 1028 nM T40097 C7NDK6 118146979 IC50 = 1249 nM T40097 C56EHT 118146984 IC50 = 653 nM T40097 CSTQ14 118716751 IC50 = 11400 nM T40097 C3R5DA 118720654 IC50 = 138 nM T40097 CGFD93 118720657 IC50 = 4495 nM T40097 C8L9SK 118720658 IC50 = 1873 nM T40097 C81HTM 118720659 IC50 = 2756 nM T40097 CC4OF9 118725553 IC50 = 970 nM T40097 CR9ML7 118725554 IC50 = 109 nM T40097 CG9Q1H 121320416 IC50 = 1670 nM T40097 CI6R3E 122178086 IC50 > 10000 nM T40097 CFD0W1 122178087 IC50 = 5100 nM T40097 CRUE70 122178088 IC50 = 318 nM T40097 CX80LD 122178090 IC50 = 3480 nM T40097 CMG2E7 122178091 IC50 = 40 nM T40097 CQ0F5Z 122178092 IC50 = 438 nM T40097 CBAQ26 127037931 IC50 = 16140 nM T40097 CMZ4C0 127037932 IC50 = 6730 nM T40097 CHJ54F 127038292 IC50 = 2770 nM T40097 CP6LM2 127038293 IC50 = 910 nM T40097 CWA51O 127038294 IC50 = 3340 nM T40097 CC6O9E 127038946 IC50 > 23000 nM T40097 CP8UX1 127039331 IC50 > 23000 nM T40097 CHC07Q 127039332 IC50 = 7170 nM T40097 CYF5A6 127039333 IC50 = 2480 nM T40097 C3QB7F 127039334 IC50 > 23000 nM T40097 CMSI81 127039335 IC50 = 18940 nM T40097 CHPR60 127039584 IC50 > 23000 nM T40097 CAN96F 127039592 IC50 > 23000 nM T40097 C4ENT5 127039909 IC50 = 19320 nM T40097 CCOM74 127040001 IC50 > 23000 nM T40097 CV82OS 127040253 IC50 > 23000 nM T40097 CDZI12 127040335 IC50 > 23000 nM T40097 C4RA8L 127040336 IC50 = 14920 nM T40097 CJSI78 127040337 IC50 > 23000 nM T40097 CAP39L 127040338 IC50 > 23000 nM T40097 CPRJ37 127040595 IC50 > 23000 nM T40097 C3UDL7 127040669 IC50 = 27070 nM T40097 CM3CJ2 127040670 IC50 > 23000 nM T40097 C7F8UR 127040991 IC50 = 6750 nM T40097 C7WZX5 127040992 IC50 > 23000 nM T40097 CH12YX 127041317 IC50 > 23000 nM T40097 C6I7UX 127041318 IC50 > 23000 nM T40097 CG6C8L 127041568 IC50 > 23000 nM T40097 C1R7IF 127041569 IC50 > 23000 nM T40097 CDO98M 127041570 IC50 > 23000 nM T40097 CK2S9X 127041849 IC50 > 23000 nM T40097 CL9YJ0 127041871 IC50 > 23000 nM T40097 C6TBN0 127041880 IC50 > 23000 nM T40097 CGBY29 127042189 IC50 > 23000 nM T40097 C87PSV 127042550 IC50 = 10930 nM T40097 C6V0QX 127042853 IC50 = 3790 nM T40097 C48VJQ 127042854 IC50 > 23000 nM T40097 CW0KG6 127042855 IC50 = 19100 nM T40097 C0FM1R 130196825 IC50 = 4171 nM T40097 C6OXE3 132134663 IC50 >= 1000 nM T40097 CTJ48K 135524085 IC50 = 960 nM T40097 CUT1W7 135524168 IC50 = 4000 nM T40097 CG9AT0 135678113 IC50 > 10000 nM T40097 CM3UC9 135883136 IC50 > 100000 nM T40097 CM2UH4 135894362 IC50 > 1000 nM T40097 CY19DW 135894364 IC50 > 1000 nM T40097 CM17FU 136198654 IC50 > 10000 nM T40097 C15HQK 136218656 IC50 > 1000 nM T40097 CZ06UK 136218660 IC50 > 1000 nM T40097 CML48X 136218661 IC50 > 1000 nM T40097 COB69I 136218662 IC50 > 1000 nM T40097 CSL6Q8 136218663 IC50 > 1000 nM T40097 CTFJ83 136226213 IC50 > 1000 nM T40097 C5EV8A 136240902 IC50 > 1000 nM T40097 CX9LB5 136240903 IC50 > 1000 nM T40097 CMC58H 136240944 IC50 > 1000 nM T40097 C60PRZ 136241012 IC50 > 1000 nM T40097 C1Q9YN 136252259 IC50 > 1000 nM T40097 C5ADF0 136252684 IC50 = 73000 nM T40097 CI1E8V 137634241 IC50 = 2670 nM T40097 CZ9BN4 138320062 IC50 = 0.032 nM T40097 C3W4RO 138403252 IC50 = 830000 nM T40097 C6VB3O 145925651 IC50 >= 5000 nM T40097 CW3RV1 145953992 IC50 = 7943.28 nM T40097 CCL34O 145954234 IC50 = 199.53 nM T40097 C4ZH8E 145954241 IC50 = 630.96 nM T40097 CNT8O5 145954713 IC50 = 158.49 nM T40097 CB0F7N 145955167 IC50 = 251.19 nM T40097 CJDG56 145960632 IC50 = 19952.62 nM T40097 CB7TW3 145960672 IC50 = 199.53 nM T40097 CH6G1S 145960935 IC50 = 316.23 nM T40097 C6ZJQ4 145961055 IC50 = 630.96 nM T40097 CZO6T7 145961089 IC50 = 1584.89 nM T40097 CX6T3J 145961172 IC50 > 10000 nM T40097 C54ZQA 145961234 IC50 = 5011.87 nM T40097 C83FPK 145961240 IC50 = 1000 nM T40097 C31QBE 145961348 IC50 = 1995.26 nM T40097 CE21QP 145961382 IC50 > 10000 nM T40097 CQ9FN7 145961544 IC50 = 1995.26 nM T40097 COCG81 145961565 IC50 = 3162.28 nM T40097 C73MVW 145961583 IC50 = 3162.28 nM T40097 C23GXR 145961663 IC50 = 79.43 nM T40097 C6HB9M 145961899 IC50 > 10000 nM T40097 CJ0K8Z 145962062 IC50 = 630.96 nM T40097 CV0T1U 145962184 IC50 = 63.1 nM T40097 CA2RO4 145962531 IC50 = 1995.26 nM T40097 CCL79I 145963000 IC50 = 125.89 nM T40097 CLFQ85 145963006 IC50 = 398.11 nM T40097 CI0V8W 145963248 IC50 > 10000 nM T40097 CYZ14S 145963250 IC50 > 10000 nM T40097 CAD5Q9 145963302 IC50 > 10000 nM T40097 C0JX1P 145963398 IC50 = 6309.57 nM T40097 C35ZRP 145963416 IC50 = 3162.28 nM T40097 CJZ4G3 145963549 IC50 = 630.96 nM T40097 C9V6AQ 145963687 IC50 = 158.49 nM T40097 CI1VH9 145985185 IC50 > 200000 nM T40097 CGZ76S 145986724 IC50 = 170 nM T40097 CNLH48 145988888 IC50 = 93600 nM T40097 CRT48W 145993502 IC50 = 88900 nM T40097 C2MD1Q 155513187 IC50 > 10000 nM T40097 CFV10S 155529132 IC50 = 820 nM T40097 CV1J4P 44576548 IC50 = 21.98 nM T40097 D00HVA 11624601 Ki = 2 nM T40097 D01HCO 23647240 IC50 = 2300 nM T40097 D02PVB 8515 IC50 = 40 nM T40097 D03UUO 23647246 IC50 = 2600 nM T40097 D06LJL 9916282 IC50 > 100000 nM T40097 D06PJW 25182616 IC50 = 5010 nM T40097 D07ADX 54764565 IC50 = 3200 nM T40097 D07HNL 23647245 IC50 = 300 nM T40097 D08IOV 1897784 IC50 = 1900 nM T40097 D08LYB 5166 IC50 > 50 nM T40097 D08UVX 23647253 IC50 = 34 nM T40097 D09PTP 57325421 IC50 = 112 nM T40097 D0E8KF 824661 IC50 = 750 nM T40097 D0F5BY 11507052 IC50 = 2100 nM T40097 D0GT8N 5154691 IC50 = 250 nM T40097 D0H2PE 10236389 IC50 > 10000 nM T40097 D0KB8D 44427133 IC50 = 700 nM T40097 D0L0HG 766949 IC50 > 10000 nM T40097 D0Q3NG 11715520 Ki = 190 nM T40097 D0S7IE 11658882 Ki = 550 nM T40097 D0SV1F 23647241 IC50 = 1100 nM T40097 D0VJ2S 57340686 IC50 = 1 nM T15797 CO92VG 11684648 IC50 = 3300 nM T15797 C1I2NF 24960729 IC50 = 440 nM T15797 C4XJ5N 78357767 IC50 > 100000 nM T15797 C94ZKU 91757965 IC50 = 2.8 nM T15797 CE5V6U 117072551 Ki = 8 nM T15797 CWM15E 118692859 IC50 = 26000 nM T15797 C30JDM 118692861 IC50 = 2200 nM T15797 CALU23 118692869 IC50 = 2400 nM T15797 C4Z9TB 118692870 IC50 = 5.6 nM T15797 CU6H8G 118692872 IC50 = 3100 nM T15797 C9F4CX 118692899 IC50 = 1400 nM T15797 C27KAV 118692924 IC50 = 5000 nM T15797 CFI1B9 118946368 IC50 > 50000 nM T15797 CVW85A 118946372 IC50 > 50000 nM T15797 C0BLZ1 121397061 IC50 = 80 nM T15797 CYX3U4 121397077 IC50 = 80 nM T15797 C5Y7VT 125407509 IC50 = 1700 nM T15797 C4D0VA 127048775 IC50 = 4200 nM T15797 CFKH80 127048776 IC50 = 50 nM T15797 CX3JL8 127049094 IC50 = 71 nM T15797 C3Z6BR 127049095 IC50 = 44 nM T15797 C9I6RY 127049096 IC50 = 19 nM T15797 CDR2I3 127049415 IC50 = 6000 nM T15797 C0VAR2 127049751 IC50 > 20000 nM T15797 C3SU0G 127049752 IC50 = 1100 nM T15797 CHS5A8 127049753 IC50 = 570 nM T15797 C4RV0W 127049754 IC50 = 38 nM T15797 C2UJ0N 127050656 IC50 = 15800 nM T15797 C2V5EI 127050657 IC50 > 20000 nM T15797 CYBO14 127050658 IC50 = 6900 nM T15797 C17CSG 127050663 IC50 = 2200 nM T15797 CXH8C5 127050664 IC50 > 20000 nM T15797 CK7U9R 127050672 IC50 = 2800 nM T15797 CF6M7Y 127050673 IC50 > 20000 nM T15797 CE80LC 127050934 IC50 > 20000 nM T15797 C2ENH5 127050971 IC50 = 8300 nM T15797 CX73BE 127050972 IC50 = 10900 nM T15797 C31MDQ 127051545 IC50 = 1700 nM T15797 C9YT7Q 127051546 IC50 = 800 nM T15797 CD2LB1 127051547 IC50 = 2200 nM T15797 C13WYM 127051858 IC50 = 119 nM T15797 CF29KH 134159782 IC50 = 62000 nM T15797 C5Q8MK 137348892 IC50 = 40 nM T15797 C5RE7T 137349288 IC50 = 8 nM T15797 C8AD4G 155514915 IC50 = 760 nM T15797 CD3S0P 155520580 IC50 = 23 nM T15797 C9MWG7 155548192 IC50 = 23 nM T15797 CZB7Y0 155555569 IC50 = 58 nM T15797 CESP32 155568735 IC50 = 32 nM T15797 D06ONB 24961094 IC50 = 120 nM T15797 D09CLP 439155 IC50 = 180 nM T15797 D0X3RK 91623361 IC50 < 15 nM T38187 CQ5VG8 44565227 EC50 = 501.19 nM T38187 CB1IO9 135407930 EC50 = 630.96 nM T38187 CX07AC 135407952 EC50 = 316.23 nM T38187 CTR26D 135407963 EC50 = 398.11 nM T38187 CQ7SZ1 135407966 EC50 = 158.49 nM T38187 C34ABJ 136036237 EC50 = 1258.93 nM T38187 C8Y7FX 136036261 EC50 = 1995.26 nM T07766 D04LVK 57379345 IC50 > 10000 nM T07766 D03LWG 53235510 IC50 > 10000 nM T07766 D07EHV 44814409 IC50 > 10000 nM T07766 D08MHM 25227462 IC50 = 190 nM T07766 D0E3TC 44259 IC50 = 1 nM T07766 D0T3ME 156422 IC50 > 30000 nM T07766 C7SFI1 10296883 IC50 > 10000 nM T07766 CACS26 11561968 Ki > 2000 nM T07766 CU0E8O 11690457 Ki > 2000 nM T07766 CB0AP2 11705863 Ki > 10000 nM T07766 C9TU1O 16046126 IC50 > 1000 nM T07766 CKR57M 16086104 IC50 > 25000 nM T07766 C16NRY 16086114 IC50 > 25000 nM T07766 CGC34R 16118737 IC50 > 25000 nM T07766 CL81VC 21100709 IC50 = 100000 nM T07766 C8NA4L 53384644 IC50 > 30000 nM T07766 C1MR8Q 60097495 IC50 > 1000 nM T07766 CV63UL 67240318 IC50 > 10000 nM T07766 C12DPO 68060125 IC50 = 39.5 nM T07766 CQC0R5 68181954 IC50 = 970 nM T07766 C82YNL 70934541 IC50 = 12.8 nM T07766 CT7V2J 71529158 IC50 = 133 nM T07766 C83FVQ 71557891 Ki = 48 nM T07766 CRX81Q 71575642 IC50 > 10000 nM T07766 C9YEQ2 73350469 IC50 = 244 nM T07766 CF8LD4 73356518 IC50 = 70.8 nM T07766 CJ2T9E 76332983 IC50 > 10000 nM T07766 CYHR27 91664373 Ki = 11 nM T07766 C4X7SD 122192466 IC50 > 10000 nM T07766 CTJ50H 127048386 Ki = 2 nM T07766 CBP5T0 127048728 Ki = 21 nM T07766 CZG30T 127051548 Ki = 3670 nM T07766 CFQ18V 127051549 Ki = 2300 nM T07766 C4P1UT 127052177 Ki = 9.5 nM T07766 C8AX0O 127052178 Ki = 4.6 nM T07766 CN37MB 127052179 Ki = 39 nM T07766 CE2B9V 127052180 Ki = 940 nM T07766 C8F0DQ 129909860 IC50 = 6 nM T07766 CZ7EX0 136183413 IC50 > 30000 nM T07766 C07EKN 138454794 IC50 > 10000 nM T07766 D06HVH 54613583 IC50 > 10000 nM T07766 D07ORL 73348907 IC50 = 64.1 nM T44011 D00ZFP 5870 Ki = 3 nM T44011 D02ENG 6918651 IC50 = 3341 nM T44011 D0B5HF 44476893 IC50 > 10000 nM T44011 D0L4FS 5280961 IC50 = 2210 nM T44011 D0O1ZI 25006684 IC50 > 30000 nM T44011 D0R8IU 24946280 IC50 > 30000 nM T44011 D0DK4I 4534 IC50 = 5500 nM T44011 CI9SZ2 3224 IC50 = 48250 nM T44011 CE82ON 92895 Ki = 24000 nM T44011 C7JEN0 94320 IC50 = 18800 nM T44011 C5A9TH 188971 Ki = 4080 nM T44011 CE18DF 317611 IC50 = 19000 nM T44011 C7HME8 439246 IC50 = 4960 nM T44011 CKB57V 440624 IC50 = 207 nM T44011 CZ0AH3 638278 IC50 = 2830 nM T44011 C2KCS3 667696 IC50 > 1000 nM T44011 CZUG74 821913 IC50 = 4800 nM T44011 CQ2GS3 2950639 IC50 = 20200 nM T44011 CZDB43 5282074 IC50 = 1090 nM T44011 CP69KZ 5324349 IC50 = 49 nM T44011 CXV6Z7 5470876 IC50 = 4100 nM T44011 C9PO8Y 6874186 IC50 = 5700 nM T44011 CPT5Y6 6918663 IC50 = 52 nM T44011 C91OZC 9879324 IC50 = 89 nM T44011 CV15NU 9953823 IC50 = 37 nM T44011 C0EO6V 10330806 IC50 = 3700 nM T44011 CXZ93W 10498888 IC50 = 790 nM T44011 CK53QH 11098954 IC50 = 109 nM T44011 C8Y1NE 11196876 IC50 = 30 nM T44011 C6K7GH 11206862 IC50 = 1700 nM T44011 CH85OD 11319723 IC50 > 30000 nM T44011 C0A7XK 11339805 IC50 = 27 nM T44011 C35FYS 11436350 IC50 = 15600 nM T44011 CA90VB 11493223 IC50 = 140 nM T44011 CN3W8L 11493379 IC50 = 85 nM T44011 C0RK4E 11500319 IC50 = 148 nM T44011 CIL69J 11515312 IC50 = 35 nM T44011 C0L8CO 11520458 IC50 = 310 nM T44011 C8NP4Y 11526147 IC50 = 2.2 nM T44011 CV3U7F 11530377 IC50 = 233 nM T44011 C6FG3C 11551133 IC50 = 633 nM T44011 C6UN3E 11565856 IC50 = 545 nM T44011 CUZ79A 11571162 IC50 = 140 nM T44011 CCZ5R4 11573293 IC50 = 121 nM T44011 CGQ5M2 11587774 IC50 = 77 nM T44011 C7XI5Y 11599989 IC50 = 93 nM T44011 C3FJQ8 11602375 IC50 = 7700 nM T44011 C2DJO8 11609517 IC50 = 32 nM T44011 CB04UF 11616864 IC50 = 320 nM T44011 C93ZPL 11616990 IC50 = 87 nM T44011 CR9L3U 11617341 IC50 = 218 nM T44011 C7CP2F 11621606 IC50 = 430 nM T44011 C3ES6U 11631931 IC50 = 73 nM T44011 C18FSY 11637932 IC50 = 10000 nM T44011 C9MD3U 11639289 IC50 = 56 nM T44011 C6OUW7 11639661 IC50 = 15 nM T44011 CW10HT 11682274 IC50 = 47 nM T44011 C5GXY7 11690058 IC50 = 123 nM T44011 CNI6C7 11700170 IC50 = 6900 nM T44011 C4LI9Y 11709431 IC50 = 392 nM T44011 C4WC9D 11710272 IC50 = 14 nM T44011 C1LQW9 11716781 IC50 = 101 nM T44011 C8X1QW 11717031 IC50 = 126 nM T44011 C2I3HX 11721764 IC50 = 120 nM T44011 CWGF07 11721794 IC50 = 1000 nM T44011 C3TYL0 11813984 IC50 = 13500 nM T44011 C2XW0P 11853305 IC50 > 30000 nM T44011 C2XRT9 16721115 IC50 > 5000 nM T44011 CG5Q4I 21043856 IC50 = 460 nM T44011 CXU49P 21157477 IC50 = 33000 nM T44011 CY9B5M 21257907 IC50 = 173 nM T44011 C79IPR 24205614 Ki = 12750 nM T44011 CE95WV 24970356 IC50 = 26 nM T44011 CM2Y8O 24995496 IC50 = 2900 nM T44011 CLZJ74 24995497 IC50 = 2000 nM T44011 CW4X9V 24995499 IC50 = 4700 nM T44011 CX5L7P 24995814 IC50 = 5400 nM T44011 CMH41V 25069448 IC50 = 36 nM T44011 CJSN68 25069763 IC50 = 33 nM T44011 CAN19S 25069766 IC50 = 70 nM T44011 CYZ9G1 25069768 IC50 = 15 nM T44011 CZ9CG8 25073248 IC50 = 14 nM T44011 CG17PN 25073557 IC50 = 12 nM T44011 C4ETA9 25073558 IC50 = 49 nM T44011 C8Z7TK 25073560 IC50 = 74 nM T44011 CL3E9G 25073863 IC50 = 28 nM T44011 C2F0MC 25074165 IC50 = 46 nM T44011 C1F9GC 25074166 IC50 = 396 nM T44011 CBRM65 25074167 IC50 = 53 nM T44011 C2P6UT 25093376 IC50 > 1000 nM T44011 CPU54X 25093388 IC50 > 5000 nM T44011 C7XZE5 25093395 IC50 > 1000 nM T44011 C2QSX4 25093396 IC50 > 1000 nM T44011 CGR64D 25192478 IC50 = 56 nM T44011 CFD5T1 25192479 IC50 = 38 nM T44011 C5SJY2 25192481 IC50 = 523 nM T44011 CPS96J 25192622 IC50 = 143 nM T44011 C62POF 39845450 IC50 = 18000 nM T44011 C5MF9Y 44189694 IC50 = 52 nM T44011 CU02PL 44314270 Ki = 59000 nM T44011 CQ3PG6 44314513 Ki = 65000 nM T44011 CX43UA 44314514 Ki = 2800 nM T44011 CV7NG0 44403805 IC50 = 730 nM T44011 CO6U7R 44403816 IC50 = 1850 nM T44011 CY8Q3U 44403818 IC50 = 950 nM T44011 CCV0T5 44403826 IC50 = 2300 nM T44011 CU8LN7 44403833 IC50 = 780 nM T44011 C2O7YQ 44403836 IC50 = 880 nM T44011 CZ3I0K 44403837 IC50 = 300 nM T44011 CQAC46 44403843 IC50 = 180 nM T44011 C02CLT 44403846 IC50 = 2750 nM T44011 COR5T8 44403850 IC50 = 920 nM T44011 C3CQ5O 44403851 IC50 = 530 nM T44011 C5CK8G 44405125 IC50 = 90 nM T44011 CO91JZ 44407474 IC50 = 460 nM T44011 CTF1O8 44422488 IC50 = 170 nM T44011 CQ1NU0 44452108 IC50 = 1800 nM T44011 COP91H 44452165 IC50 = 3700 nM T44011 CC41MD 44452190 IC50 = 8300 nM T44011 C79MED 44452239 IC50 = 9900 nM T44011 C12BET 44452272 IC50 = 3700 nM T44011 C1MP4N 44456578 IC50 = 171 nM T44011 CH82JM 44456599 IC50 = 44 nM T44011 C6HTI5 44542044 IC50 > 5000 nM T44011 C2P6FA 44542045 IC50 > 1000 nM T44011 C04CHV 44542193 IC50 = 130 nM T44011 C2K6RE 44542194 IC50 = 29 nM T44011 CH61ZI 44542650 IC50 > 5000 nM T44011 CZY93O 44542651 IC50 > 1000 nM T44011 C3ZSO6 44542652 IC50 > 5000 nM T44011 CTO1G9 44542799 IC50 > 1000 nM T44011 CG81LA 44542947 IC50 > 5000 nM T44011 C0Q2NE 44542948 IC50 > 5000 nM T44011 CJDR60 44543104 IC50 = 427 nM T44011 C1R7PN 44543105 IC50 = 620 nM T44011 C0RG9O 44543108 IC50 = 17 nM T44011 C2T6KW 44561552 IC50 = 47000 nM T44011 C1N9JI 44585930 IC50 = 1320 nM T44011 CBP1V8 44585931 IC50 = 840 nM T44011 C8TD2A 45484071 IC50 = 350 nM T44011 C1AF4H 46879677 IC50 = 193 nM T44011 C1Z9UX 49840059 IC50 = 22 nM T44011 C7W5AR 49840060 IC50 = 368 nM T44011 C9VSY7 49840061 IC50 = 945 nM T44011 CR1U5L 49840062 IC50 = 33 nM T44011 C37JRZ 49840063 IC50 = 95 nM T44011 C3RND0 49840065 IC50 = 21 nM T44011 CVM0N8 49840128 IC50 = 46 nM T44011 CWV8K1 49840129 IC50 = 18 nM T44011 C1AZW7 49840130 IC50 = 594 nM T44011 CIV03C 49840131 IC50 = 207 nM T44011 C4A0MP 49840132 IC50 = 30 nM T44011 C9G8JM 49840133 IC50 = 6 nM T44011 CRYC81 49840134 IC50 = 8 nM T44011 C8V2DY 49840135 IC50 = 17 nM T44011 CG15NJ 49840195 IC50 = 16 nM T44011 CS39TD 49840196 IC50 = 126 nM T44011 CSZL58 49840197 IC50 = 86 nM T44011 C8OQK6 49840198 IC50 = 108 nM T44011 CZ1AV0 49840200 IC50 = 20 nM T44011 CC4HY7 49840201 IC50 = 199 nM T44011 CA8N9P 52911994 IC50 > 100000 nM T44011 C1N6AB 53317188 IC50 = 510 nM T44011 C38PYT 53317908 IC50 = 8516 nM T44011 C0SP1Q 53319802 IC50 = 4300 nM T44011 CAUB79 53319854 IC50 = 810 nM T44011 CJAD87 53322150 IC50 = 1000 nM T44011 C3DE5X 53323495 IC50 = 420 nM T44011 CEZ97N 53323760 IC50 = 1500 nM T44011 CO9DF6 53324805 IC50 = 1150 nM T44011 C8XC7R 53325844 IC50 = 614 nM T44011 CXJ34L 53326359 IC50 = 380 nM T44011 CQ95PJ 53326449 IC50 = 290 nM T44011 CQU5D6 53326823 IC50 = 27 nM T44011 C9H5YE 53361128 IC50 > 10000 nM T44011 CL7K5O 53494954 IC50 = 68 nM T44011 CGH4U1 53863164 IC50 = 44 nM T44011 CGY29J 56643459 IC50 = 611 nM T44011 C25QVY 56648121 IC50 = 1748 nM T44011 C5LW3H 56648217 IC50 = 919 nM T44011 C0Q2LX 56648219 IC50 = 2245 nM T44011 C0T5LQ 56648221 IC50 = 713 nM T44011 CA6XQ8 56648223 IC50 = 309 nM T44011 CQR86G 56648305 IC50 = 926 nM T44011 CT5F7P 56648307 IC50 = 1130 nM T44011 C7A6ZL 56649596 IC50 = 4452 nM T44011 C31HUC 56680365 IC50 = 1000 nM T44011 CKY51C 56847605 IC50 = 27 nM T44011 CQ93RT 56928979 IC50 = 12 nM T44011 C58IXP 56929075 IC50 = 8 nM T44011 CZRQ14 56929159 IC50 = 13 nM T44011 CD65YQ 56929161 IC50 = 136 nM T44011 CVNH50 56929162 IC50 = 38 nM T44011 C5ZBY7 56929246 IC50 = 863 nM T44011 CA14UJ 56929248 IC50 = 99 nM T44011 C90URY 56929249 IC50 = 11 nM T44011 CR75VG 56929252 IC50 = 152 nM T44011 CC7YI5 56929343 IC50 = 243 nM T44011 C9NIE8 56929344 IC50 = 3000 nM T44011 CZ91ML 56929345 IC50 = 171 nM T44011 CT71OR 56929346 IC50 = 667 nM T44011 CU5PI9 56929436 IC50 = 29 nM T44011 C6D3AR 56933761 IC50 > 100000 nM T44011 CQD1G4 56933896 IC50 = 13009 nM T44011 C8SRA4 56933897 IC50 > 100000 nM T44011 C7OM3Q 56933898 IC50 = 64532 nM T44011 CUN84A 56933900 IC50 = 9099 nM T44011 CT3K8N 56933902 IC50 = 3801 nM T44011 CFV1S4 56934037 IC50 > 10000 nM T44011 CG26KN 56934038 IC50 = 5449 nM T44011 C8I6GS 56934039 IC50 > 120000 nM T44011 CJBG32 56934040 IC50 = 5105 nM T44011 CUF4M8 56934042 IC50 = 2982 nM T44011 CCP9X6 56934182 IC50 = 3915 nM T44011 C5X4YJ 56934183 IC50 > 100000 nM T44011 CRG9O0 56934185 IC50 > 100000 nM T44011 C2QI1L 56934187 IC50 = 55741 nM T44011 CYO56W 56934188 IC50 > 100000 nM T44011 CT09PY 56934323 IC50 = 43398 nM T44011 CN24XA 56934324 IC50 > 40000 nM T44011 CIT84G 56934325 IC50 = 23345 nM T44011 CBGF96 56934326 IC50 = 18597 nM T44011 C6FDS7 56934327 IC50 = 10645 nM T44011 CIC42E 56934328 IC50 = 3151 nM T44011 C1L2UV 56934478 IC50 = 18040 nM T44011 CNB3O1 56934479 IC50 = 202 nM T44011 CID83Q 56969690 IC50 = 475 nM T44011 CK1OW6 56969691 IC50 = 413 nM T44011 C9IWR5 56969692 IC50 = 2429 nM T44011 C98EFI 56969693 IC50 = 1764 nM T44011 CA18ZV 56969694 IC50 = 571 nM T44011 CW8B5N 56969897 IC50 = 289 nM T44011 C8AB6T 56969898 IC50 = 53 nM T44011 CYFM98 56969899 IC50 = 159 nM T44011 C8SJM5 56969902 IC50 = 5480 nM T44011 CN5E3O 56969903 IC50 = 1272 nM T44011 CE0YB8 56969904 IC50 = 1013 nM T44011 C9RTC7 57384260 IC50 = 29 nM T44011 CKOJ47 57384261 IC50 = 22 nM T44011 C2PVF3 57384262 IC50 = 53 nM T44011 CR9M5S 57384263 IC50 = 701 nM T44011 CV6I9E 57384264 IC50 = 19 nM T44011 C85QLG 57384514 IC50 = 31 nM T44011 CMI40L 57384515 IC50 = 33 nM T44011 CK1W2U 57384516 IC50 = 633 nM T44011 CA03RF 57384517 IC50 = 32 nM T44011 CF23UZ 57384518 IC50 = 32 nM T44011 CJGY80 57384781 IC50 = 519 nM T44011 CC7IH1 57387800 IC50 = 92 nM T44011 C9P3JU 57388026 IC50 = 196 nM T44011 C6EAS2 57388027 IC50 = 17 nM T44011 CEMR25 57388028 IC50 = 690 nM T44011 C5M9TB 57388029 IC50 = 21 nM T44011 C6WT9D 57388030 IC50 = 25 nM T44011 C39SNL 57916360 IC50 > 35000 nM T44011 CN6Z5E 60165269 IC50 > 50000 nM T44011 CCPV67 60196493 IC50 = 6728 nM T44011 CG0VN3 60196497 IC50 = 4337 nM T44011 C8N5EK 60196599 IC50 = 6217 nM T44011 C7Y2SN 60196600 IC50 = 1927 nM T44011 CC68DY 60196601 IC50 = 10573 nM T44011 CR4TP3 60196604 IC50 > 40000 nM T44011 CH75LW 60196703 IC50 = 5306 nM T44011 C84EMK 60196704 IC50 = 6752 nM T44011 CQ5FE7 60196705 IC50 = 4812 nM T44011 C5Z3UD 60196706 IC50 = 5426 nM T44011 CQI2U6 60196810 IC50 = 11454 nM T44011 C2WMG3 60196811 IC50 = 6800 nM T44011 CV0R9D 60196812 IC50 = 8209 nM T44011 C56WAS 60196815 IC50 = 12259 nM T44011 C0HG7E 60196905 IC50 = 1109 nM T44011 C96JBP 60196908 IC50 = 4821 nM T44011 C9J4FK 60196910 IC50 = 18663 nM T44011 C2TPB9 60197003 IC50 = 85343 nM T44011 C9REP6 60197921 IC50 > 60000 nM T44011 C2T6CV 71450526 Ki = 69400 nM T44011 CR0EZ7 71454153 Ki = 424500 nM T44011 C6IVL9 71455202 IC50 = 221 nM T44011 C0RT9Z 71455718 IC50 = 430 nM T44011 CJO0A2 71456991 IC50 = 13 nM T44011 C1TJ3D 71458857 IC50 = 5 nM T44011 CNR8P0 73346456 IC50 = 2031 nM T44011 C2N3DX 73346458 IC50 = 4299 nM T44011 CHR94D 73347958 IC50 = 238 nM T44011 C8XY1B 73347959 IC50 = 3282 nM T44011 CRAT17 73354019 IC50 = 427 nM T44011 CJ8QD3 73357097 IC50 = 1308 nM T44011 CD1C5J 76321189 IC50 = 172 nM T44011 C2KEA0 76335656 IC50 = 153 nM T44011 C29IZS 90645097 IC50 = 22298 nM T44011 CRL96S 90645098 IC50 = 1641 nM T44011 CG0T9C 90645099 IC50 = 984 nM T44011 CR7W4I 90645100 IC50 = 3071 nM T44011 C41WAJ 90645101 IC50 = 3096 nM T44011 CDT4A0 90645102 IC50 = 2485 nM T44011 C02WYL 90645103 IC50 = 432 nM T44011 CGLB58 90645104 IC50 = 336 nM T44011 CV1U6X 90645568 IC50 = 90 nM T44011 C4I5XD 90645569 IC50 = 157 nM T44011 C0XF9A 90645570 IC50 = 120 nM T44011 C1T5GV 90645571 IC50 = 152 nM T44011 CO1WI3 90645572 IC50 = 104 nM T44011 CB7LV8 90645573 IC50 = 275 nM T44011 CPA10J 90645574 IC50 = 752 nM T44011 CA01SR 90645575 IC50 = 630 nM T44011 COW3D0 91820627 IC50 = 0.2 nM T44011 C6FQ8M 118714402 IC50 = 195 nM T44011 C1GU9B 118714405 IC50 = 89 nM T44011 CSP23C 118716517 IC50 = 4306 nM T44011 CQWD38 118716518 IC50 = 3825 nM T44011 CH91QY 118716519 IC50 = 4570 nM T44011 CQNM84 118716520 IC50 = 1177 nM T44011 CVNC84 118716521 IC50 = 698 nM T44011 CG60CE 118716523 IC50 = 2687 nM T44011 CSA17F 118716524 IC50 = 1562 nM T44011 CLNK01 118716526 IC50 = 11576 nM T44011 CG2I5V 118716527 IC50 = 9412 nM T44011 C8ADE4 118716528 IC50 = 2144 nM T44011 CK7Z1A 118716532 IC50 = 25302 nM T44011 CN7SK0 118716537 IC50 = 11541 nM T44011 CO13JK 118716544 IC50 = 16732 nM T44011 CX62KM 118733245 IC50 = 6600 nM T44011 C9EN3B 118733250 IC50 = 1400 nM T44011 CFDE04 122194299 IC50 = 145 nM T44011 C38UXF 122194300 IC50 = 195 nM T44011 C3E8JV 122194301 IC50 = 169 nM T44011 CIN2J9 122194302 IC50 = 151 nM T44011 CF8L9B 122194303 IC50 = 21 nM T44011 CW2C9S 122194304 IC50 = 23 nM T44011 C7Q5CR 122194305 IC50 = 39 nM T44011 CR7IL2 122194306 IC50 = 16 nM T44011 C0A1VC 122194307 IC50 = 33 nM T44011 C0XR5H 122194308 IC50 = 71 nM T44011 C01MKU 122194309 IC50 = 56 nM T44011 CB17CP 122194310 IC50 = 32 nM T44011 CJB07W 122194311 IC50 = 47 nM T44011 CK23IP 122194312 IC50 = 42 nM T44011 C2X5BZ 122194313 IC50 = 182 nM T44011 C9DFZ7 122194314 IC50 = 50 nM T44011 CD2GK1 122194315 IC50 = 38 nM T44011 C7SK8P 122194316 IC50 = 30 nM T44011 CR94NZ 122194317 IC50 = 50 nM T44011 C1A6RY 122194318 IC50 = 109 nM T44011 CPED85 122194319 IC50 = 135 nM T44011 CLS5U7 122194320 IC50 = 35 nM T44011 CN7FY8 122194321 IC50 = 311 nM T44011 CSN0Z1 122194322 IC50 = 17 nM T44011 C2N6OQ 122194406 IC50 = 18 nM T44011 CJM82P 122194407 IC50 = 51 nM T44011 CHK61C 122194408 IC50 = 112 nM T44011 C4SE0C 122194409 IC50 = 10 nM T44011 COLZ59 122194410 IC50 = 2 nM T44011 CE59LP 122194411 IC50 = 3 nM T44011 CYXJ37 122194412 IC50 = 2 nM T44011 CH4FI6 122194413 IC50 = 4 nM T44011 CG2U4J 122194414 IC50 = 6 nM T44011 CGL35E 122194415 IC50 = 2 nM T44011 CU95PH 122194416 IC50 = 5 nM T44011 C6PBV0 122194417 IC50 = 5 nM T44011 C73DYS 122194418 IC50 = 38 nM T44011 CW4HZ0 122194419 IC50 = 12 nM T44011 C3A9SE 122652894 IC50 = 0.5 nM T44011 CK13ZA 122652897 IC50 = 48 nM T44011 C6O0JQ 122652898 IC50 = 0.4 nM T44011 CXM0P4 122652900 IC50 = 55 nM T44011 C6HG7D 122652901 IC50 = 49 nM T44011 C8JTM5 122652904 IC50 = 7.3 nM T44011 CU46WZ 122652905 IC50 = 8 nM T44011 CZ7FA6 122652912 IC50 = 30 nM T44011 CZU8P4 122652913 IC50 = 3.3 nM T44011 C3L4RF 122652915 IC50 = 1.2 nM T44011 CD6L0M 122652921 IC50 = 3.3 nM T44011 C08DFN 122652926 IC50 = 7 nM T44011 CHQ67B 122652928 IC50 = 92 nM T44011 C6QEY9 122652929 IC50 = 21 nM T44011 C6WM7D 122652930 IC50 = 15 nM T44011 C37CQE 122652932 IC50 = 76 nM T44011 CTUZ47 122652933 IC50 = 0.9 nM T44011 C2Q8AK 122652936 IC50 = 0.3 nM T44011 CK7X2Q 122652942 IC50 = 4.7 nM T44011 CX1EM2 122652943 IC50 = 44 nM T44011 CJ0NE8 122652945 IC50 = 0.9 nM T44011 CV0H7E 122652946 IC50 = 0.4 nM T44011 CJ27FT 122652947 IC50 = 150 nM T44011 C2LD0O 122652950 IC50 = 2.1 nM T44011 CFDR29 122652951 IC50 = 6 nM T44011 CQB51Y 122652955 IC50 = 59 nM T44011 CL2A9J 122652956 IC50 = 235 nM T44011 CCG94B 122652957 IC50 = 6 nM T44011 C0WE5T 122652958 IC50 = 1.3 nM T44011 CFB94G 122652962 IC50 = 7 nM T44011 CLYR93 122652963 IC50 = 2.1 nM T44011 C3MF5K 122652969 IC50 = 5.8 nM T44011 CA7QT5 122652970 IC50 = 1.7 nM T44011 CXE43V 122652972 IC50 = 3.1 nM T44011 C0YHG5 122652975 IC50 = 27 nM T44011 C68ONT 122652976 IC50 = 6.8 nM T44011 CD4Z0J 122652979 IC50 = 21 nM T44011 CD27AG 122652981 IC50 = 4.7 nM T44011 C95QKJ 122652982 IC50 = 10 nM T44011 C19JRB 122652985 IC50 = 6.7 nM T44011 C8JT3D 122652987 IC50 = 84 nM T44011 C0KDG2 122652990 IC50 = 4.8 nM T44011 CTZS18 122652994 IC50 = 1.2 nM T44011 CZ68HG 122652995 IC50 = 15 nM T44011 C57QKX 122652996 IC50 = 96 nM T44011 C3AH2K 122652997 IC50 = 5.9 nM T44011 CC7UI6 122652998 IC50 = 0.5 nM T44011 C7CT4F 122653001 IC50 = 150 nM T44011 C1RIK0 122653002 IC50 = 0.5 nM T44011 C9G4NV 122653003 IC50 = 1.4 nM T44011 CI7C2T 122653005 IC50 = 27 nM T44011 C2B7ZX 122653009 IC50 = 49 nM T44011 CNK06Z 122653011 IC50 = 2.4 nM T44011 CRO6V0 122653012 IC50 = 130 nM T44011 C5D8UG 122653014 IC50 = 13 nM T44011 CC5KH8 122653016 IC50 = 1.5 nM T44011 C4NZP0 122653018 IC50 = 5.2 nM T44011 CG8A2U 122653030 IC50 = 18 nM T44011 CR9Y4L 122653033 IC50 = 3.5 nM T44011 C1VZ3I 122653039 IC50 = 53 nM T44011 C2EIB6 122653041 IC50 = 2.4 nM T44011 C2NBH7 122653046 IC50 = 35 nM T44011 CY3JD6 122660686 IC50 = 3400 nM T44011 COD0A4 122660687 IC50 = 47 nM T44011 CY3X6R 122660690 IC50 = 105 nM T44011 CXQ0H1 122660691 IC50 = 899 nM T44011 C3HA5L 127038736 IC50 = 16100 nM T44011 CH30BC 127038737 IC50 = 26300 nM T44011 C3FAU0 127038740 IC50 = 9600 nM T44011 CKX3B8 127040395 IC50 = 13300 nM T44011 CD2H6A 127042310 IC50 = 60100 nM T44011 CHQ5A1 135567209 IC50 = 22395 nM T44011 CJZ1N9 135899471 IC50 > 1000 nM T44011 C2HN4U 135899472 IC50 > 5000 nM T44011 CQBT39 135899489 IC50 = 413 nM T44011 C6XAB4 135955190 IC50 = 64 nM T44011 CFR38I 136042244 IC50 = 567 nM T44011 C7PCS0 136042245 IC50 = 19650 nM T44011 CP65AH 136042246 IC50 = 60638 nM T44011 CFRW24 136168827 IC50 = 78 nM T44011 C1M3US 136183444 IC50 = 35 nM T44011 C25XTW 137632454 IC50 = 7.1 nM T44011 C3G1SO 137636708 IC50 = 10.2 nM T44011 CNB52O 137638205 IC50 = 1.1 nM T44011 C2V5JX 137639781 IC50 = 18 nM T44011 C1FDY3 137640192 IC50 = 1.4 nM T44011 CBE4K2 137640293 IC50 = 3 nM T44011 C7OHY5 137643959 IC50 = 22.5 nM T44011 CSB8P0 137644465 IC50 = 6 nM T44011 C5FP6M 137645395 IC50 = 43.5 nM T44011 CE0OK4 137646056 IC50 = 32.4 nM T44011 CEXP59 137646742 IC50 = 73 nM T44011 C3IKG5 137647263 IC50 = 11 nM T44011 C8U2DH 137649984 IC50 = 3.4 nM T44011 CFU3V9 137652166 IC50 = 2.2 nM T44011 CPKR15 137656256 IC50 = 12.2 nM T44011 CB06TQ 137660131 IC50 = 20 nM T44011 C62FZT 137661419 IC50 = 2.7 nM T44011 C41SYN 139030522 IC50 = 45.8 nM T44011 CH35RO 145982486 IC50 = 5.3 nM T44011 CHGR75 145985839 IC50 = 50 nM T44011 C8R4ZF 145990266 IC50 = 35 nM T44011 C4NUH3 145992326 IC50 = 27 nM T44011 C9WK4M 145993875 IC50 = 27 nM T44011 C6E4ZP 155513937 IC50 = 4.6 nM T44011 C6R2WG 155514963 IC50 = 198 nM T44011 CE37TP 155515038 IC50 = 1.2 nM T44011 CKQY72 155515127 IC50 = 17.2 nM T44011 CP46TY 155516583 IC50 = 4.3 nM T44011 CC8AD1 155516734 IC50 = 2.3 nM T44011 CPN6I1 155519849 IC50 = 10.1 nM T44011 C1P3IC 155523432 IC50 = 170 nM T44011 CY2SA5 155525017 IC50 = 6.3 nM T44011 CK5YJ7 155526302 IC50 = 0.1 nM T44011 C5O2TK 155526475 IC50 = 306 nM T44011 CJ4WH6 155527207 IC50 = 3.9 nM T44011 CD2Y9X 155527324 IC50 = 15.6 nM T44011 C6UI1F 155528716 IC50 = 7.2 nM T44011 CS5F3D 155529123 IC50 = 45.4 nM T44011 C9M7DU 155530633 IC50 = 0.8 nM T44011 C8TBY3 155531966 IC50 = 0.6 nM T44011 C4K3GZ 155534601 IC50 = 11.4 nM T44011 C1IC7Z 155535276 IC50 = 6.9 nM T44011 CO0E9Z 155537294 IC50 = 5 nM T44011 CGN69L 155538884 IC50 = 3.9 nM T44011 CH6Y0B 155542289 IC50 = 8.2 nM T44011 C20UFI 155544948 IC50 = 8 nM T44011 C87PHQ 155545568 IC50 = 0.1 nM T44011 CVS93D 155548405 IC50 = 3 nM T44011 COQ8P0 155548975 IC50 = 1.7 nM T44011 CDEY45 155553373 IC50 = 0.7 nM T44011 C9K6RV 155558001 IC50 = 2 nM T44011 C3IH4O 155560831 IC50 = 80 nM T44011 C9RH3F 155562009 IC50 = 8.8 nM T44011 CM6EX7 155562215 IC50 = 1.4 nM T44011 CQBJ79 155564096 IC50 = 20.3 nM T44011 CXZ9Q6 155564371 IC50 = 3.1 nM T44011 D00PSW 3630776 IC50 = 7.5 nM T44011 D00PUR 46887555 IC50 = 1370 nM T44011 D00RIX 5280443 IC50 = 710 nM T44011 D00SLE 25093373 IC50 = 50 nM T44011 D00YNA 25093374 IC50 = 243 nM T44011 D01AVM 53319855 IC50 = 300 nM T44011 D01JVG 44542048 IC50 = 42 nM T44011 D01KKU 5281894 IC50 = 5250 nM T44011 D01RZP 25192621 IC50 = 64 nM T44011 D01ZCG 25093386 IC50 = 69 nM T44011 D02BEJ 44542795 IC50 = 780 nM T44011 D02UUR 135855877 IC50 = 1610 nM T44011 D03BZT 12985714 IC50 = 340 nM T44011 D03XHF 44542049 IC50 = 113 nM T44011 D05AIT 46887580 IC50 = 1390 nM T44011 D06CED 46844318 IC50 = 560 nM T44011 D07JOZ 44542195 IC50 = 123 nM T44011 D07VXQ 25093398 IC50 = 101 nM T44011 D08OKP 25192476 IC50 = 402 nM T44011 D08OQX 25093392 IC50 = 185 nM T44011 D08PDK 24950391 IC50 = 40 nM T44011 D09GQE 25192619 IC50 = 629 nM T44011 D0A2GN 25192480 IC50 = 535 nM T44011 D0A4XA 25093379 IC50 = 169 nM T44011 D0A7PU 46887581 IC50 = 850 nM T44011 D0B6SF 44542047 IC50 = 493 nM T44011 D0BF3Y 44543260 IC50 = 51 nM T44011 D0C9KZ 25093397 IC50 = 471 nM T44011 D0DC3E 25093399 IC50 = 1000 nM T44011 D0EL1Y 24857878 IC50 = 310 nM T44011 D0F6ZH 12316406 IC50 = 2257 nM T44011 D0G1DN 25093384 IC50 = 342 nM T44011 D0G3TK 5280863 IC50 = 1050 nM T44011 D0G5CP 46887511 IC50 = 690 nM T44011 D0H8PI 10308021 IC50 = 2425 nM T44011 D0I5YT 25093391 IC50 = 77 nM T44011 D0IZ4Z 25192184 IC50 = 1850 nM T44011 D0J8LU 44543257 IC50 = 171 nM T44011 D0M0KX 25192477 IC50 = 8 nM T44011 D0M3RQ 24827431 IC50 = 1232 nM T44011 D0NM0P 25093389 IC50 = 151 nM T44011 D0P6JE 44543261 IC50 = 567 nM T44011 D0P8PK 10192730 IC50 = 116 nM T44011 D0Q3AN 44543255 IC50 = 64 nM T44011 D0Q6AD 46887551 IC50 = 1020 nM T44011 D0QX5D 46887579 IC50 = 2380 nM T44011 D0R3HP 269792 IC50 = 201 nM T44011 D0R5WV 21861202 IC50 = 336 nM T44011 D0T6WL 25093377 IC50 = 455 nM T44011 D0TA0J 25093387 IC50 = 173 nM T44011 D0UR6C 25192620 IC50 = 717 nM T44011 D0V2QH 24894072 IC50 = 20 nM T44011 D0W5CR 446201 Ki = 3 nM T44011 D0Y2RL 25192475 IC50 = 46 nM T44011 D0Z1MJ 44542800 IC50 = 119 nM T40000 D07XHO 4413 IC50 = 650 nM T40000 D0FT4R 107706 IC50 > 2000 nM T40000 D0Y6SQ 2536 IC50 = 1480 nM T40000 D03QJN 9895762 Ki = 61 nM T40000 D0N7WR 108040 Ki = 610 nM T40000 CLX4V7 130395 IC50 = 2320 nM T40000 C1BHS3 193409 Ki = 23000 nM T40000 CZP0Y1 204101 Ki > 2300 nM T40000 C5QKC3 448605 Ki = 40 nM T40000 CX5MS1 448610 Ki = 1000 nM T40000 C8I0VG 5289529 Ki = 14000 nM T40000 C2ZRF5 6540265 Ki > 10000 nM T40000 CN57IY 6540268 Ki > 100000 nM T40000 C8OE6S 6913584 IC50 = 190 nM T40000 C4VX9Y 9803558 IC50 > 10000 nM T40000 C4OTK6 9805415 IC50 = 5800 nM T40000 C6JIT7 9806444 IC50 > 11000 nM T40000 CS1DL7 9826716 IC50 = 250 nM T40000 CB82VS 9827306 IC50 > 11000 nM T40000 CGN48U 9827867 IC50 > 2500 nM T40000 C5Z2RH 9848091 IC50 > 11000 nM T40000 CIL85V 9871029 IC50 > 11000 nM T40000 C6ZB3K 9872552 IC50 > 11000 nM T40000 C1M2PU 9892103 IC50 > 11000 nM T40000 C1C3VT 9914538 IC50 > 11000 nM T40000 C5KS0R 9936020 IC50 > 11000 nM T40000 C49DRC 9936691 IC50 > 11000 nM T40000 C0R4GE 9954812 IC50 = 2100 nM T40000 C2Y0QV 9959268 IC50 = 2100 nM T40000 CFQV59 10007890 IC50 > 10000 nM T40000 CEN06H 10093642 IC50 = 96.5 nM T40000 C3TWI1 10095455 Ki > 100000 nM T40000 C5E0SY 10126451 Ki = 525 nM T40000 CS2G4T 10140847 Ki = 19 nM T40000 C12USI 10146294 Ki = 810 nM T40000 C7L5IJ 10157296 Ki = 265 nM T40000 CL7U8P 10181581 Ki = 295 nM T40000 CEP79T 10216518 Ki = 206 nM T40000 C8V1AY 10225952 Ki = 69 nM T40000 C0J1TD 10278414 Ki = 100 nM T40000 CNAX45 10287785 Ki = 336 nM T40000 C5EDW1 10294146 Ki = 400 nM T40000 CMNP39 10389039 IC50 > 10000 nM T40000 CEH4D1 10391881 Ki > 10000 nM T40000 CLK08Z 10391999 IC50 > 10000 nM T40000 CD0VI1 10412365 Ki > 10000 nM T40000 CU8N3V 10578280 Ki > 1000000 nM T40000 CEJ14F 10624997 Ki > 1000000 nM T40000 CPWH69 10648370 Ki > 1000000 nM T40000 CBT96N 10664145 Ki > 10000000 nM T40000 CW1G9B 10672666 IC50 = 86 nM T40000 CGYR23 10696955 Ki > 1000000 nM T40000 C3IN8W 10815545 Ki > 1000000 nM T40000 CVQE76 10816339 Ki > 1000000 nM T40000 CW7Q2U 10895700 IC50 > 10000 nM T40000 C91GMZ 11317532 Ki > 100000 nM T40000 CIQH43 11445130 IC50 = 240 nM T40000 CVI82D 11479420 Ki > 2300 nM T40000 CJP9O1 11684611 Ki = 650 nM T40000 CNPW05 11755188 IC50 > 10000 nM T40000 CPR4I1 12047383 Ki = 87000 nM T40000 C5U0FJ 12047384 Ki = 87000 nM T40000 C5FU3H 12047385 Ki = 45000 nM T40000 CPB09W 13192674 IC50 = 25700 nM T40000 CO0J3T 13192685 IC50 = 36000 nM T40000 CY87AI 14488960 IC50 = 33300 nM T40000 CM8W7C 14488962 IC50 = 11200 nM T40000 C6VM2S 14488964 IC50 = 19000 nM T40000 CK5Z7P 14488966 IC50 = 20300 nM T40000 C7EIL0 14488968 IC50 = 25600 nM T40000 C50XDQ 14488970 IC50 = 14800 nM T40000 C54JLM 14488972 IC50 = 29300 nM T40000 C0WSE1 14488974 IC50 = 82400 nM T40000 CH9I4M 14488976 IC50 = 11800 nM T40000 C5CK1E 14488978 IC50 = 53800 nM T40000 C37MRI 16718808 IC50 > 10000 nM T40000 CO2JG4 20595081 IC50 > 11000 nM T40000 CM7BH1 20595091 IC50 > 11000 nM T40000 CCH5N1 20595225 IC50 > 11000 nM T40000 C2ID8R 20595260 IC50 > 10000 nM T40000 CMT46A 20595328 IC50 > 10000 nM T40000 CIM9C3 20801121 Ki > 10000 nM T40000 CC1Y0R 20801139 Ki > 10000 nM T40000 CS3HB4 20801160 Ki > 100000 nM T40000 CNTI15 21366511 IC50 > 11000 nM T40000 C5S8ZW 21366513 IC50 > 11000 nM T40000 C67QCO 21366574 IC50 > 11000 nM T40000 CS2L1Y 21366575 IC50 > 11000 nM T40000 CX1WM9 21366579 IC50 > 11000 nM T40000 CA63IO 21706943 Ki = 3300 nM T40000 C80JYP 21707001 Ki = 3700 nM T40000 C3H6XW 21707065 Ki = 2482 nM T40000 C5JD2U 21707080 Ki = 1900 nM T40000 CN6P9I 22394409 Ki = 8540 nM T40000 C3TOL6 23106311 IC50 = 39810.72 nM T40000 C1L9VZ 23647194 Ki > 10000 nM T40000 CC29KT 23647198 Ki > 10000 nM T40000 CVO5L6 24748791 IC50 = 1370 nM T40000 COX4A7 24873356 Ki = 25 nM T40000 C2H4PJ 25166809 Ki > 30000 nM T40000 CL7NY5 44274017 IC50 = 9700 nM T40000 CMG90C 44274089 IC50 > 10000 nM T40000 C8Y9JZ 44284991 Ki > 63 nM T40000 CMZ71H 44284992 Ki = 120 nM T40000 C5NU9L 44285118 Ki = 160 nM T40000 CU9G2F 44285211 Ki = 9.5 nM T40000 C0FPN1 44285253 Ki = 34 nM T40000 C9N1ZL 44285281 Ki > 4.3 nM T40000 C5PX3O 44285312 Ki = 9.5 nM T40000 C9LRW8 44285352 Ki = 370 nM T40000 C0DG5R 44287043 Ki = 92000 nM T40000 CZRH12 44290033 IC50 > 11000 nM T40000 CUY95P 44290108 IC50 > 11000 nM T40000 CL0U1A 44303806 IC50 = 3162.28 nM T40000 C7BO3I 44314289 Ki = 31 nM T40000 CZQ3V4 44314305 Ki = 21 nM T40000 C8KOM9 44333945 Ki > 150000 nM T40000 CH32DA 44333955 Ki > 2500000 nM T40000 C75KOP 44333957 Ki > 50000 nM T40000 C7A6KF 44333986 Ki = 7000 nM T40000 CF1LQ4 44333999 Ki = 223000 nM T40000 CZ7RK3 44334001 Ki = 191000 nM T40000 CUO4N2 44334160 Ki = 47300 nM T40000 C7Y8IG 44334488 Ki = 70 nM T40000 CHL01I 44334805 Ki = 300 nM T40000 CRT4G3 44335601 Ki > 1000000 nM T40000 C7Z9WL 44335624 Ki > 1000000 nM T40000 CXL2Q8 44341827 Ki = 199000 nM T40000 CAY27D 44392382 Ki = 640 nM T40000 C2SQ1C 44392401 Ki = 992 nM T40000 C4VKE9 44392403 Ki = 42 nM T40000 CYL52J 44392413 Ki = 54 nM T40000 CN8CJ3 44392416 Ki = 379 nM T40000 CE42KB 44392423 Ki = 156 nM T40000 CORK28 44392427 Ki = 1402 nM T40000 C30CFX 44436704 IC50 = 820 nM T40000 CW5V7Y 44559839 Ki = 3600 nM T40000 C0Y7GN 53736009 IC50 = 6309.57 nM T40000 CPBW48 57392333 Ki = 1300000 nM T40000 CL2JE5 57395841 Ki = 1800000 nM T40000 CTE30K 57842560 Ki = 22 nM T40000 C0C6UB 57842624 Ki = 100 nM T40000 C7XY5A 57842673 Ki = 18 nM T40000 CU9S6K 57842710 Ki = 6 nM T40000 CL8T7M 57842742 Ki = 35 nM T40000 C41NSR 57842812 Ki = 1900 nM T40000 C9XW1C 57842830 Ki = 4700 nM T40000 CWF0C3 57842850 Ki = 100 nM T40000 C73CPB 57842913 Ki = 100 nM T40000 CM8UJ7 57976444 Ki = 1200 nM T40000 CQ71KE 57976446 Ki > 30000 nM T40000 CPW2H7 59315536 Ki = 2900 nM T40000 CO38AC 59402011 Ki > 30000 nM T40000 CE5A7B 60162406 Ki > 50000 nM T40000 CZN12D 70691542 Ki = 31 nM T40000 CCO4X9 71455264 Ki = 50 nM T40000 C40BMT 71455265 Ki = 110 nM T40000 CHBA35 71462441 Ki = 8 nM T40000 CJPF90 71548883 Ki > 10000 nM T40000 C30ZKJ 71561420 Ki = 10000 nM T40000 C78DJQ 71711730 IC50 < 10000 nM T40000 CM83VP 72163524 IC50 > 10000 nM T40000 CK34ZH 72550138 Ki = 650 nM T40000 CDA91I 72550584 Ki = 100 nM T40000 CT45ER 72550807 Ki = 390 nM T40000 C46TNC 72550811 Ki = 600 nM T40000 CXM6C2 72550813 Ki = 1100 nM T40000 CLI36U 72551247 Ki = 650 nM T40000 C1MBU7 72793747 IC50 > 50000 nM T40000 C6BY5D 72793776 IC50 > 50000 nM T40000 C1DI8A 72793778 IC50 > 50000 nM T40000 C60JSR 73353029 Ki = 630000 nM T40000 CD8M1N 73354683 IC50 = 32400 nM T40000 C5U9CI 73355715 Ki = 0.0049 nM T40000 CIN46O 86343959 Ki = 140 nM T40000 CWS28P 86344699 Ki = 9.4 nM T40000 CWP85J 87360663 IC50 > 10000 nM T40000 C65TLW 101862198 Ki > 1000000 nM T40000 C28PCL 117749867 Ki = 23 nM T40000 C3PS6Y 118098650 Ki = 270 nM T40000 C5E8QD 118098664 Ki = 790 nM T40000 C0GRU4 118718129 Ki = 6.1 nM T40000 C3YVQ8 122164611 Ki = 1150 nM T40000 CY1S5D 122164612 Ki = 1200 nM T40000 CK0W2P 127027635 Ki > 30000 nM T40000 CJ6DA9 127028140 IC50 > 2500 nM T40000 CD9KI3 127028141 IC50 > 2500 nM T40000 C1BWV2 127035672 Ki = 384 nM T40000 CVRY56 127036086 Ki = 201 nM T40000 C9B6LT 127037264 Ki = 833 nM T40000 C60HLK 127037469 Ki > 1000000 nM T40000 C4T9KU 127045502 Ki = 4 nM T40000 C4RFP7 127045503 Ki = 31 nM T40000 C2IOG9 127045504 Ki = 154 nM T40000 CHK80O 127045505 Ki = 25 nM T40000 CL6W5N 127045506 Ki = 36 nM T40000 CPQ04R 134132204 Ki = 21 nM T40000 CC7UO1 134133660 Ki = 5300 nM T40000 C9USR6 134134113 IC50 = 12600 nM T40000 C34AJF 134137014 IC50 = 400000 nM T40000 C18WFV 134140132 Ki = 110 nM T40000 C6DPW7 134141496 Ki = 580 nM T40000 C5WC3I 134143793 IC50 = 221000 nM T40000 CIRU10 134145163 Ki = 200 nM T40000 CHA7X9 134146314 Ki = 260 nM T40000 CLW95Y 134146409 Ki = 3100 nM T40000 COF6A2 134147357 Ki > 100000 nM T40000 C9UZI0 134148669 Ki = 15 nM T40000 CTG65U 134148771 Ki = 34 nM T40000 CR6V9U 134150310 Ki = 960 nM T40000 CUW75P 134151146 IC50 = 125000 nM T40000 C3QEO5 134151811 Ki = 2600 nM T40000 CG9UL4 134156593 Ki = 1600 nM T40000 COJ20R 137322719 IC50 = 316.23 nM T40000 CDQ62V 137637214 Ki > 50000 nM T40000 C2K8JV 137639385 Ki = 50000 nM T40000 CNX46H 137654508 Ki > 50000 nM T40000 CUZ35A 138115400 IC50 = 63095.73 nM T40000 CAG81E 155511419 IC50 > 6309.57 nM T40000 CZR36C 155511554 IC50 = 316227.77 nM T40000 CV5F4A 155511614 IC50 = 79432.82 nM T40000 C1GYM7 155513506 IC50 = 3981.07 nM T40000 C4IZX3 155514387 IC50 = 63095.73 nM T40000 CMY9P0 155514527 IC50 = 25118.86 nM T40000 CW2X7K 155514934 IC50 = 50118.72 nM T40000 C0OY1S 155518519 IC50 = 7943.28 nM T40000 C6NX4K 155519661 IC50 = 398.11 nM T40000 C4MS1B 155519676 IC50 > 10000 nM T40000 CT4L1S 155520177 IC50 > 50118.72 nM T40000 CG2WM9 155520998 IC50 = 630957.34 nM T40000 C41TFK 155521732 IC50 = 1258.93 nM T40000 C49DMZ 155522189 IC50 = 79432.82 nM T40000 CLM04O 155522595 IC50 = 15848.93 nM T40000 CIH95K 155523037 IC50 = 199526.23 nM T40000 C2KM7D 155524369 IC50 = 1995.26 nM T40000 C0MUB5 155525046 IC50 > 10000 nM T40000 CSPB43 155525076 IC50 = 3162.28 nM T40000 COT61Y 155526156 IC50 = 10000 nM T40000 CIPV21 155526440 IC50 > 5011.87 nM T40000 CXBR96 155526691 IC50 = 158489.32 nM T40000 CN3BH5 155527998 IC50 > 10000 nM T40000 CHYW65 155528639 IC50 >= 6309.57 nM T40000 CKW0N3 155528746 IC50 = 63095.73 nM T40000 CD7O2G 155530095 IC50 > 10000 nM T40000 C42LDK 155530603 IC50 = 79432.82 nM T40000 C35QWO 155531023 IC50 = 1995.26 nM T40000 CENG47 155531694 IC50 = 10000 nM T40000 CIH96R 155532277 IC50 = 31622.78 nM T40000 C9CH2J 155532630 IC50 = 501187.23 nM T40000 CG03WZ 155533183 IC50 = 50118.72 nM T40000 CC2TH3 155534011 IC50 = 12589.25 nM T40000 C3R0PV 155535171 IC50 > 5011.87 nM T40000 C12HON 155536142 IC50 > 10000 nM T40000 C7RBN1 155536236 IC50 = 5011.87 nM T40000 CVCN73 155539549 IC50 = 79432.82 nM T40000 CR3HF2 155539807 IC50 = 12589.25 nM T40000 CYQ5N7 155540505 IC50 = 398107.17 nM T40000 C0IXU7 155540672 IC50 = 630.96 nM T40000 CY6DK3 155540964 IC50 = 1584.89 nM T40000 C2PL7Y 155541127 IC50 = 19952.62 nM T40000 C97IBT 155542437 IC50 = 39810.72 nM T40000 CHYZ70 155544016 IC50 = 125.89 nM T40000 CX9A5M 155547612 IC50 = 25118.86 nM T40000 C5MB9R 155547962 IC50 = 630.96 nM T40000 CG8F4S 155548359 IC50 = 5011.87 nM T40000 CLFB25 155548371 IC50 > 10000 nM T40000 C75CKY 155550727 IC50 = 31622.78 nM T40000 COM52R 155551892 IC50 >= 3981.07 nM T40000 CJ3FI5 155553630 IC50 > 10000 nM T40000 CMV2T0 155553751 IC50 = 39810.72 nM T40000 C5BH7C 155553819 IC50 = 6309.57 nM T40000 C9BKN7 155554975 IC50 = 6309.57 nM T40000 CSW48V 155557718 IC50 = 251.19 nM T40000 CFZ8Y9 155557932 IC50 = 501.19 nM T40000 CNOI61 155558524 IC50 = 501187.23 nM T40000 C6D8KL 155560348 IC50 = 158489.32 nM T40000 CZI5S1 155563470 IC50 = 25118.86 nM T40000 CM8XB1 155565537 IC50 = 31622.78 nM T40000 C8N3SP 155566632 IC50 = 251.19 nM T40000 CAK16X 155566796 IC50 = 501187.23 nM T40000 CN6BS0 155567190 IC50 > 2511.89 nM T40000 CIU2C9 155568927 IC50 = 12589.25 nM T40000 D00POF 21707121 Ki = 991 nM T40000 D06AVE 10200844 Ki = 576 nM T40000 D0A8WP 447732 Ki = 2500 nM T40000 D0J2SM 296008 IC50 = 9890 nM T40000 D0K0GU 44392430 Ki = 83 nM T40000 D0S4MQ 44392405 Ki = 770 nM T81623 D09JEJ 24748573 IC50 = 17 nM T81623 D0E3TC 44259 IC50 = 3.45 nM T81623 D0MS3Z 16725726 IC50 = 81 nM T81623 D03BNU 59604787 IC50 > 10000 nM T81623 D0T3ME 156422 IC50 > 30000 nM T81623 C18WEB 490561 IC50 = 360 nM T81623 CG1VY6 813906 IC50 = 529.5 nM T81623 CCGT78 1551558 IC50 = 583 nM T81623 C4J0QW 1733425 IC50 = 227.1 nM T81623 CAV19R 2360773 IC50 < 1000 nM T81623 C38JRK 2406980 IC50 = 346.1 nM T81623 CQO23Z 5285453 IC50 = 713.7 nM T81623 CJA65E 5400660 IC50 = 533.5 nM T81623 CW5C3O 5796642 IC50 = 278.5 nM T81623 C5NJ0G 5842430 IC50 = 395.3 nM T81623 C76RMA 5953789 IC50 = 148.4 nM T81623 C9XK5Y 6030124 IC50 = 157 nM T81623 CT30MZ 6187657 IC50 = 359.6 nM T81623 CLR41O 6516567 IC50 = 278.5 nM T81623 CK21EQ 9796713 IC50 > 1000 nM T81623 CJH69P 9840393 IC50 > 1000 nM T81623 CBOP58 11293798 Ki > 10000 nM T81623 C26BZX 11362471 Ki > 10000 nM T81623 CWXB93 11397177 Ki > 10000 nM T81623 CTG83F 11539329 Ki > 1400 nM T81623 CMIL86 11590363 Ki > 1400 nM T81623 C9T6SC 11640926 Ki > 1400 nM T81623 C4NO7Y 11809063 IC50 > 1000 nM T81623 CFPW41 16007116 Ki > 1400 nM T81623 C20DST 16105503 IC50 > 1000 nM T81623 CCN62F 16105510 IC50 = 487 nM T81623 C5VPH9 16129448 IC50 = 1600 nM T81623 CBO4L2 16450385 IC50 = 291.2 nM T81623 CX1HL8 25032704 Ki = 27.3 nM T81623 CY3HW5 46224684 IC50 = 4300 nM T81623 CLS29B 46872626 IC50 > 10000 nM T81623 C2O8RZ 46886323 IC50 > 1000 nM T81623 CEQN27 52936621 Ki > 1000 nM T81623 C0SWH5 53348216 IC50 > 40000 nM T81623 C8NA4L 53384644 IC50 = 32000 nM T81623 CDK93W 56946894 IC50 = 10 nM T81623 CK6WO0 66552478 IC50 < 10000 nM T81623 C37NKO 67129970 IC50 = 4860 nM T81623 CK80LJ 67130050 IC50 = 4980 nM T81623 CV63UL 67240318 IC50 > 10000 nM T81623 C7GRV2 68755406 IC50 > 10000 nM T81623 C2B4SW 118714182 IC50 = 39820 nM T81623 CJI0G1 135520135 IC50 = 700 nM T81623 CH64ID 136175114 IC50 = 1800 nM T81623 C2WP5B 136175121 IC50 = 140 nM T81623 C1TS6F 136175122 IC50 = 450 nM T81623 CB5G4X 136175123 IC50 > 10000 nM T81623 CSGM03 137210056 IC50 = 510 nM T81623 CI1E8V 137634241 IC50 > 10000 nM T81623 C4DRX1 137643187 IC50 = 12150 nM T81623 CGW9I0 137656387 IC50 = 18880 nM T81623 C2MD1Q 155513187 IC50 > 10000 nM T81623 D00ERW 44444843 Ki > 1391 nM T81623 D00HVA 11624601 Ki > 1400 nM T81623 D0GN5Z 5281295 IC50 = 2330 nM T81623 D0Q3NG 11715520 Ki > 1400 nM T81623 D0S7IE 11658882 Ki > 1400 nM T03513 D07MEH 3033769 Ki = 5.1 nM T03513 D0D1AL 3559 IC50 = 5 nM T03513 D0H6QU 6005 IC50 = 25 nM T03513 D0R9EQ 5095 EC50 = 100 nM T03513 D0T7OW 681 IC50 = 15 nM T03513 D00OWF 5280953 Ki > 10000 nM T03513 D08AWI 11430856 Ki > 2000 nM T03513 CK1JY9 3106 EC50 = 80 nM T03513 C8Y6DE 37461 IC50 = 50 nM T03513 C53TUG 132435 EC50 = 122 nM T03513 CF2JG6 156376 IC50 = 8000 nM T03513 CGT8R0 160510 Ki > 10000 nM T03513 CYV1R3 417052 Ki > 10000 nM T03513 C6AJX9 3049326 EC50 = 700 nM T03513 C9BM2I 9991512 Ki = 20 nM T03513 C5ZLK0 10060449 Ki = 57 nM T03513 C0P5WB 10067380 Ki = 159 nM T03513 CD0M9Y 10081286 EC50 = 116 nM T03513 C5PDQ8 10242850 Ki = 334 nM T03513 C2UNO6 10251160 Ki = 11 nM T03513 C5RF0W 10264090 Ki = 49 nM T03513 C57PKI 10330528 Ki = 222 nM T03513 CPK71L 10356389 Ki = 106 nM T03513 CEX1T3 10384736 Ki = 162 nM T03513 CT3DJ5 10391240 Ki = 1100 nM T03513 CS3OC4 10405678 Ki = 1736 nM T03513 C60ICT 10420915 Ki = 430 nM T03513 C4YBI9 10428654 Ki = 353 nM T03513 CS1LF0 10450580 Ki = 315 nM T03513 CIG85H 11282247 IC50 > 33000 nM T03513 CNYK74 11743212 Ki = 120 nM T03513 CZS90F 13530907 EC50 > 1000 nM T03513 CPX35V 14890801 Ki = 88.5 nM T03513 C1Y0BL 14890813 Ki = 17.3 nM T03513 C2U4VC 14890816 Ki = 41.1 nM T03513 C59WZE 15654433 Ki = 40 nM T03513 CMZ4Q9 44317801 Ki = 2610 nM T03513 CKX8V3 44317821 Ki = 130 nM T03513 CGL51N 44325577 Ki = 125 nM T03513 CXPS18 44325578 Ki = 89 nM T03513 COM07T 44325658 Ki = 21 nM T03513 C4K6BH 52946883 Ki > 10000 nM T03513 CY92LZ 53310757 Ki > 1000 nM T03513 CAB2G8 70696007 Ki = 2620 nM T03513 CVF5P0 73603034 IC50 = 500 nM T03513 C8K9XA 122196341 IC50 > 1200 nM T03513 D05TZE 133741 EC50 = 1.8 nM T03513 D0H3KU 172267 IC50 = 16 nM T46000 D0E3TC 44259 IC50 = 0.0825 nM T46000 C3VRO9 44557921 IC50 > 10000 nM T46000 CV63UL 67240318 IC50 > 10000 nM T46000 CXC69T 137321158 IC50 = 106 nM T46000 C2MD1Q 155513187 IC50 > 10000 nM T46000 D0C2GE 67161540 IC50 = 25 nM T92828 D09TBD 5344 IC50 = 24000 nM T92828 D0S7JH 16004692 IC50 = 391 nM T92828 D0U4CE 104865 Ki = 80 nM T92828 D0X5ZI 6918493 IC50 = 195 nM T92828 D08IXA 16759603 IC50 = 0.41 nM T92828 D09LQK 443289 IC50 > 1000 nM T92828 D0AW8E 151174 IC50 = 21 nM T92828 D0H2RJ 6433095 IC50 = 175 nM T92828 D0LI1C 44469321 IC50 > 30000 nM T92828 D0QG1B 25099191 IC50 = 987 nM T92828 D0R7YY 177236 IC50 = 16 nM T92828 D0Y6UU 159594 IC50 = 63.3 nM T92828 D01EDE 5311192 Ki = 1 nM T92828 D01VUE 122272 IC50 = 14000 nM T92828 D02HVW 9910224 IC50 > 100 nM T92828 D07YHT 178103 Ki = 110 nM T92828 D0B5PU 9843631 Ki = 18700 nM T92828 D0H0KK 11742628 IC50 = 4550 nM T92828 D0J2IH 9912992 IC50 = 600 nM T92828 D0J5HU 122044 IC50 = 1100 nM T92828 D0L3AR 23670447 Ki = 139 nM T92828 D0T1RG 216235 IC50 = 9.8 nM T92828 D0W6XL 108002 Ki = 14.7 nM T92828 CPTS80 123883 IC50 = 130 nM T92828 C6MRZ0 182140 IC50 > 500000 nM T92828 CLT7A1 197712 Ki = 195 nM T92828 CN01ID 345351 IC50 = 30000 nM T92828 CZN6S9 743974 EC50 > 50118.72 nM T92828 CAWU68 3370402 IC50 = 88000 nM T92828 CNIO83 3795752 IC50 = 80000 nM T92828 CM6FP0 3811690 IC50 = 14000 nM T92828 C25GEL 3921421 Ki = 230 nM T92828 CTYX34 5122650 Ki = 1900 nM T92828 CP1I9X 6433100 Ki = 7.15 nM T92828 C4UJF5 9797546 Ki > 200000 nM T92828 CSDO82 9799352 Ki > 200000 nM T92828 CUZ05W 9803428 IC50 = 7940 nM T92828 C1S4LE 9806559 IC50 = 18000 nM T92828 CL1Q0S 9807200 IC50 = 347 nM T92828 C3I8FC 9807456 IC50 = 1190 nM T92828 CT3NI6 9807691 IC50 = 380 nM T92828 CH5D6W 9808545 IC50 = 2.2 nM T92828 CA1M0Q 9809270 IC50 = 931 nM T92828 CW7DO3 9809919 IC50 = 5 nM T92828 C2OHV0 9810190 IC50 > 2500 nM T92828 CK5R3H 9810400 IC50 = 4 nM T92828 CN2R6T 9810571 IC50 = 24 nM T92828 C5SPK1 9818889 Ki > 200000 nM T92828 CF04WY 9820754 IC50 > 250000 nM T92828 C74IRJ 9821701 IC50 = 410 nM T92828 C4JI2K 9822616 Ki = 16000 nM T92828 CY6HF0 9825494 IC50 = 200 nM T92828 CE6D8F 9826741 IC50 = 5740 nM T92828 C1T8FJ 9829478 IC50 = 569 nM T92828 C5O9JC 9830098 Ki = 1200 nM T92828 CS93GB 9830495 IC50 = 33 nM T92828 CLO82B 9830773 IC50 = 122 nM T92828 CTL39M 9831249 IC50 = 2 nM T92828 C1VP5Q 9831527 IC50 = 9 nM T92828 CAE70F 9840391 IC50 = 55000 nM T92828 C5PW0N 9840650 Ki > 200000 nM T92828 C8KIE6 9845562 IC50 = 390 nM T92828 C45MZP 9846065 IC50 = 8500 nM T92828 CD7Z8S 9849547 Ki = 14.7 nM T92828 CXS8Q0 9850566 IC50 = 50 nM T92828 CY4ZL7 9852318 IC50 = 12 nM T92828 C72WKR 9852624 IC50 = 101 nM T92828 CMG10J 9853025 IC50 = 100 nM T92828 CR23PL 9853077 IC50 = 16 nM T92828 C57ROU 9853680 IC50 = 7 nM T92828 CKN2M5 9864017 Ki = 66000 nM T92828 C1DN5I 9864880 IC50 > 10000 nM T92828 CE3C9Z 9865409 Ki = 19.7 nM T92828 CX4G1B 9865706 IC50 > 25000 nM T92828 C8GX0U 9868379 IC50 = 1800 nM T92828 C2A5TY 9868822 IC50 = 1800 nM T92828 CR4E6U 9869444 IC50 = 5600 nM T92828 CZY6C2 9870830 IC50 = 120 nM T92828 C04NGY 9870959 IC50 = 14100 nM T92828 CAR36G 9871348 IC50 = 340 nM T92828 CD8UW0 9871561 IC50 = 914 nM T92828 CDN81J 9873255 IC50 = 397 nM T92828 C60BJE 9874379 IC50 = 81 nM T92828 CI6CX4 9874557 IC50 = 19 nM T92828 C41CBX 9888574 IC50 = 5200 nM T92828 CG57RJ 9890440 IC50 > 1140 nM T92828 CJ4TB6 9894443 IC50 = 6.6 nM T92828 CR4WY5 9894460 IC50 = 4.4 nM T92828 CLS9V6 9894916 IC50 > 100000 nM T92828 CB0A3I 9896251 IC50 = 60 nM T92828 CT17KX 9897092 IC50 = 4 nM T92828 CJ10PX 9897720 IC50 = 60 nM T92828 C72NYE 9909467 IC50 = 3300 nM T92828 CZ9P6O 9913198 IC50 > 2500 nM T92828 CAL58B 9914310 IC50 = 98 nM T92828 CU8H1Z 9915028 Ki = 13000 nM T92828 CQ1ZN4 9915510 IC50 = 397 nM T92828 C2Q9GB 9916121 IC50 = 3058 nM T92828 C94UCB 9916235 IC50 = 0.28 nM T92828 C5D9ZU 9917072 IC50 = 15 nM T92828 C4Z8KR 9917706 IC50 = 4 nM T92828 C2UWJ3 9927658 Ki > 200000 nM T92828 CDE9G5 9932004 IC50 = 225 nM T92828 CE3GU4 9934580 IC50 = 2000 nM T92828 CH34SZ 9936145 IC50 = 4400 nM T92828 CHY6M2 9937336 Ki = 25 nM T92828 CI3B9H 9938533 Ki = 1.2 nM T92828 C5E1FA 9938571 IC50 = 38 nM T92828 CD6CI8 9939238 IC50 = 25 nM T92828 COQ6D7 9939960 IC50 = 440 nM T92828 C5LQV8 9953358 Ki = 371 nM T92828 CYNC62 9953821 IC50 > 500000 nM T92828 C7TWX3 9955200 IC50 = 1550 nM T92828 CSXQ79 9956918 IC50 = 12200 nM T92828 CL81WX 9957225 IC50 > 25000 nM T92828 C6HL8T 9957883 IC50 = 280 nM T92828 C5VW8U 9958321 Ki = 770 nM T92828 C6HLP5 9959298 IC50 = 90000 nM T92828 C5P2DZ 9961131 IC50 = 103 nM T92828 CTZ12I 9961347 IC50 = 3.3 nM T92828 CD12UT 9979632 Ki = 24.5 nM T92828 CDSG04 9980487 IC50 > 2500 nM T92828 CHNZ10 9985589 IC50 = 3.6 nM T92828 C9UT3E 10005597 IC50 = 41 nM T92828 C6BLV3 10024044 IC50 > 2500 nM T92828 C9CS4P 10027018 IC50 > 25000 nM T92828 CU20QS 10029171 IC50 = 774 nM T92828 C7KB8D 10038537 IC50 > 25000 nM T92828 C95BSU 10045790 Ki = 757 nM T92828 C3SX8N 10047521 IC50 > 2700 nM T92828 C69CLY 10070783 IC50 = 2700 nM T92828 C2FQS4 10076527 IC50 = 571 nM T92828 CU4Y3I 10088869 Ki > 30000 nM T92828 C27QDR 10095637 IC50 = 47000 nM T92828 CCQ9E3 10096179 Ki = 344 nM T92828 CER7B9 10102342 IC50 > 10000 nM T92828 CNF2H4 10116355 IC50 = 47000 nM T92828 CS4BZ7 10119105 IC50 = 13800 nM T92828 C9EOW5 10119177 IC50 = 30 nM T92828 CE7HG5 10119517 Ki = 3360 nM T92828 C6EA9N 10120430 IC50 = 13.2 nM T92828 C1NCD2 10122033 IC50 = 202 nM T92828 CHG8V4 10122442 IC50 = 18 nM T92828 CE73TY 10122495 IC50 = 199 nM T92828 CQ35RE 10122675 IC50 = 236 nM T92828 CGK62Y 10129267 IC50 = 566 nM T92828 C6AYB1 10137382 IC50 = 8240 nM T92828 CH13YM 10138169 IC50 = 7000 nM T92828 CS9T6L 10140418 IC50 = 558 nM T92828 CKT17H 10140871 IC50 = 183 nM T92828 CU1FG6 10140965 IC50 = 16800 nM T92828 C9DQ8U 10144334 IC50 = 77 nM T92828 C4ZF9E 10144372 IC50 = 2030 nM T92828 CDJ2E1 10145418 IC50 = 465 nM T92828 CV39YI 10146305 IC50 = 100 nM T92828 CIL90P 10146377 IC50 = 241 nM T92828 C0XP7T 10146640 IC50 = 42 nM T92828 C9H2YW 10151203 IC50 = 6800 nM T92828 C6DV9U 10160887 IC50 = 4500 nM T92828 CP6S8W 10163956 IC50 = 65.6 nM T92828 C4R9AN 10165809 IC50 = 612 nM T92828 CYMP81 10166139 IC50 = 15.5 nM T92828 CLT63F 10166543 IC50 = 83.6 nM T92828 C8S2OA 10166981 IC50 = 47.1 nM T92828 CHS67I 10168195 IC50 = 366 nM T92828 CF9A4T 10168597 IC50 = 920 nM T92828 CG47TJ 10168939 IC50 = 1060 nM T92828 CN1DM8 10173807 IC50 = 120 nM T92828 CYLB74 10184817 IC50 = 71000 nM T92828 CRQ3M8 10185233 IC50 = 744 nM T92828 C15RSN 10187261 IC50 = 21.4 nM T92828 CMN3L6 10187313 IC50 = 109 nM T92828 CA84YS 10187997 IC50 = 0.6 nM T92828 CSI1V8 10188517 IC50 = 50 nM T92828 CE9K4V 10189776 IC50 = 973 nM T92828 CZ3QV1 10190108 IC50 = 123 nM T92828 C3RM1T 10195727 IC50 = 1600 nM T92828 CW73GD 10205245 IC50 = 40400 nM T92828 CG53PL 10205429 IC50 = 2880 nM T92828 C4V8OE 10209814 IC50 = 49.7 nM T92828 CQ5PU8 10210086 IC50 = 1030 nM T92828 CX37UN 10210629 IC50 = 0.48 nM T92828 C3W0LP 10211543 IC50 = 207 nM T92828 C17TGP 10211772 IC50 = 589 nM T92828 C4D2OL 10211781 IC50 = 197 nM T92828 C2XQ5M 10212088 IC50 = 28 nM T92828 C1PA3X 10212163 IC50 = 1400 nM T92828 C3Z0YT 10216862 IC50 = 2700 nM T92828 CA9IR4 10218058 IC50 = 1131 nM T92828 C05NBT 10224228 IC50 = 18100 nM T92828 C4JN9U 10224745 IC50 = 184 nM T92828 CEH63U 10226215 IC50 = 35500 nM T92828 C9E5VZ 10226239 IC50 = 250 nM T92828 CM9X1P 10230375 IC50 > 10000 nM T92828 C2V3IA 10230546 IC50 = 22.4 nM T92828 CHE0D9 10230703 IC50 = 48.1 nM T92828 C5XB6S 10230737 IC50 = 17.7 nM T92828 CA2M7S 10231591 IC50 = 49 nM T92828 C1AQ8P 10233400 IC50 = 656 nM T92828 C1W7CZ 10238141 IC50 = 940 nM T92828 CRT27P 10240093 IC50 = 460 nM T92828 CYVT16 10244529 IC50 > 25000 nM T92828 C0V1MY 10265127 IC50 = 57000 nM T92828 CZXR27 10274552 IC50 = 34300 nM T92828 CV0W4U 10275056 IC50 = 8160 nM T92828 CO18IK 10278777 IC50 = 62000 nM T92828 CGN2Z4 10279940 IC50 = 25700 nM T92828 C09UWV 10281192 IC50 = 205 nM T92828 C2MYV8 10281573 IC50 = 44 nM T92828 CQG29F 10281606 IC50 = 832 nM T92828 CS4H7T 10281943 IC50 = 1140 nM T92828 CQ2DL1 10282008 IC50 = 32.2 nM T92828 CEH24R 10282163 IC50 = 221 nM T92828 CS5QZ1 10288713 IC50 = 450 nM T92828 CD93FM 10289311 IC50 = 64000 nM T92828 C9HT0L 10289348 IC50 = 95000 nM T92828 C6TO5E 10298354 IC50 = 108 nM T92828 CE2IN9 10299975 IC50 = 8000 nM T92828 C64KQN 10302118 IC50 = 1520 nM T92828 CE8O1S 10303258 IC50 = 11.1 nM T92828 C5FD9N 10303311 IC50 = 70.3 nM T92828 C56YUP 10304227 IC50 = 1670 nM T92828 C57EVT 10305181 IC50 = 603 nM T92828 C3IQ9D 10305334 IC50 = 32 nM T92828 CQN59O 10310877 IC50 = 1200 nM T92828 CY1O3L 10321290 IC50 = 11 nM T92828 C4HD5U 10321341 Ki = 1044 nM T92828 CZDC58 10342643 IC50 = 1750 nM T92828 CV05AX 10344511 IC50 = 1720 nM T92828 CL32JM 10344914 IC50 = 62 nM T92828 CN5F3X 10346184 IC50 = 2670 nM T92828 CVBP57 10347080 IC50 = 275 nM T92828 CQVP17 10347783 IC50 = 565 nM T92828 CNP9A3 10357554 IC50 = 49000 nM T92828 CM12GP 10364227 IC50 = 400 nM T92828 CV9W0K 10366278 IC50 = 42 nM T92828 CFQ31T 10366742 IC50 = 2910 nM T92828 CKB78T 10383884 IC50 = 930 nM T92828 CY8TH3 10391487 IC50 = 5080 nM T92828 CEOA37 10407051 Ki = 2443 nM T92828 CRJ63P 10410546 IC50 > 2500 nM T92828 C2YZ6V 10412464 IC50 > 2500 nM T92828 CB24TQ 10426645 IC50 = 4900 nM T92828 CJ2Z1I 10429404 IC50 = 5200 nM T92828 CG3FC5 10432263 Ki = 20.4 nM T92828 C2T8QW 10433234 IC50 = 6600 nM T92828 C2FIW7 10453858 Ki = 483 nM T92828 CNOP08 10463627 IC50 = 590 nM T92828 C4VE7N 10477792 IC50 > 500000 nM T92828 C4R6AL 10478562 IC50 = 23000 nM T92828 CG4SX2 10479787 IC50 = 2090 nM T92828 CQFV65 10501279 IC50 = 12000 nM T92828 CJ6N8I 10502226 IC50 = 27200 nM T92828 CG3PQ2 10502577 IC50 = 10100 nM T92828 CA28OV 10503067 IC50 = 1300 nM T92828 CTN0R4 10503334 IC50 = 77600 nM T92828 CE6O4M 10503525 IC50 = 640 nM T92828 CL15XB 10503921 IC50 = 3900 nM T92828 CVD26B 10503976 IC50 > 100000 nM T92828 CYSG24 10504542 IC50 = 7410 nM T92828 C8N3GD 10504689 IC50 = 6000 nM T92828 CWI0N5 10504920 IC50 = 25700 nM T92828 C2DFV1 10505209 IC50 = 16000 nM T92828 CB31YK 10505357 Ki = 320 nM T92828 CST2V6 10505434 Ki = 170 nM T92828 C6ZV2G 10505771 IC50 = 8000 nM T92828 CJFM87 10506068 IC50 > 2500 nM T92828 CKE8Q4 10506430 IC50 = 5.8 nM T92828 CC6GL2 10506505 IC50 > 100000 nM T92828 CIW27H 10508342 Ki = 215 nM T92828 CEG80Q 10525281 IC50 = 17400 nM T92828 COH58N 10526002 IC50 > 2500 nM T92828 C4KPF8 10527706 IC50 = 4570 nM T92828 CPD1A6 10527774 IC50 = 67400 nM T92828 CRYH40 10528383 IC50 = 15400 nM T92828 CGL8S2 10528863 Ki = 16.2 nM T92828 C57AKG 10529742 IC50 = 43600 nM T92828 C7H8QX 10529868 IC50 = 4 nM T92828 C9VB4O 10530409 IC50 = 260 nM T92828 C6VMG1 10531506 IC50 = 31 nM T92828 CN3K9V 10546830 IC50 > 100000 nM T92828 C2L5NQ 10548486 IC50 = 67600 nM T92828 CH3TX0 10548722 Ki = 78000 nM T92828 CGJ98W 10549472 Ki = 110000 nM T92828 C5PBZ2 10550033 IC50 > 100000 nM T92828 CV60OA 10552007 IC50 = 1600 nM T92828 CL7X5F 10552051 IC50 > 100000 nM T92828 C5GH9V 10552413 IC50 = 26200 nM T92828 CM30IW 10552548 IC50 = 2200 nM T92828 C9SW8J 10552683 Ki = 1300 nM T92828 CV7R5Z 10552883 IC50 = 10000 nM T92828 C6RH4Q 10553165 IC50 = 5400 nM T92828 CDLU05 10553384 IC50 = 42000 nM T92828 CMW5I1 10553490 IC50 = 14400 nM T92828 CIE84N 10553793 Ki = 115 nM T92828 CBY05M 10554085 IC50 > 100000 nM T92828 CSVQ94 10554273 IC50 > 100000 nM T92828 CT5JP4 10554384 IC50 > 100000 nM T92828 C4BSH1 10554410 IC50 > 100000 nM T92828 CUTR43 10554539 IC50 = 15800 nM T92828 CID50O 10555112 Ki = 24 nM T92828 C2BDQ5 10555191 IC50 > 2500 nM T92828 CGF3D2 10555208 IC50 = 3.4 nM T92828 C1RS0J 10555424 IC50 = 2100 nM T92828 CL20OW 10555806 IC50 = 0.71 nM T92828 C8GL9N 10575755 IC50 > 100000 nM T92828 C29LIN 10575845 IC50 = 51900 nM T92828 C49SNK 10576377 IC50 = 63100 nM T92828 C69OHR 10576378 IC50 = 61700 nM T92828 C7ES1R 10576379 IC50 = 30200 nM T92828 CT75CF 10576427 IC50 = 880 nM T92828 CLW2T1 10576863 IC50 > 2500 nM T92828 C9NS2G 10576888 IC50 = 19500 nM T92828 C4C7XI 10576889 IC50 = 117000 nM T92828 CB5Q2P 10576910 IC50 = 33200 nM T92828 C38AFS 10577255 IC50 = 6170 nM T92828 C8FJ5L 10577306 IC50 > 100000 nM T92828 C0MC2P 10577388 IC50 = 82 nM T92828 C6BKQ7 10577405 IC50 = 36000 nM T92828 CI0AM1 10577829 IC50 = 62000 nM T92828 CCNG64 10577879 IC50 > 2500 nM T92828 C94LZB 10578300 IC50 > 100000 nM T92828 CFJ4B1 10578601 IC50 > 100000 nM T92828 C8BK7V 10578853 IC50 = 600 nM T92828 C8YF3Z 10579100 IC50 = 47 nM T92828 CN20UM 10579885 IC50 > 2500 nM T92828 CEM46W 10597575 IC50 = 630 nM T92828 CW4NU5 10599129 Ki = 1000 nM T92828 CV69ID 10599230 IC50 = 579 nM T92828 CRM76K 10599879 IC50 = 9120 nM T92828 CHD87J 10600668 IC50 = 4500 nM T92828 CX25TC 10601668 IC50 = 850 nM T92828 CL5Q1J 10602183 IC50 = 41000 nM T92828 C2I0VP 10602267 IC50 = 85000 nM T92828 CM83DC 10602451 IC50 > 100000 nM T92828 CKA92J 10602620 IC50 = 82 nM T92828 CK2F0S 10602743 IC50 = 180 nM T92828 CN1KQ0 10603135 Ki = 160 nM T92828 C3C6ZP 10603409 IC50 = 0.14 nM T92828 C9YZD4 10604119 IC50 = 1.7 nM T92828 C46ZEW 10604167 IC50 = 744 nM T92828 CPEL02 10604797 IC50 > 2500 nM T92828 C3M5OI 10615322 IC50 > 100000 nM T92828 C7GCV1 10621170 IC50 = 92100 nM T92828 CSLD54 10622380 IC50 = 19100 nM T92828 CR0A3H 10622616 IC50 > 2500 nM T92828 CO80EG 10623877 IC50 = 17000 nM T92828 CY0K7C 10624645 Ki = 55 nM T92828 CIU5B9 10625152 IC50 = 26000 nM T92828 CKZ31J 10625269 IC50 = 74 nM T92828 C7H1BX 10625270 IC50 = 16 nM T92828 CA0C8T 10625694 IC50 = 2.6 nM T92828 C9QFT0 10625738 IC50 = 8710 nM T92828 CH40JY 10626031 IC50 > 100000 nM T92828 C74JIT 10626177 IC50 > 90000 nM T92828 C4GPV2 10626245 IC50 = 79000 nM T92828 CJW2V0 10626362 IC50 = 0.94 nM T92828 C0CR7L 10626646 IC50 = 460 nM T92828 CNQ73U 10627272 IC50 = 200 nM T92828 C5XGP4 10627805 IC50 = 10 nM T92828 CB6O1X 10645550 IC50 > 2500 nM T92828 C8E5AX 10646372 IC50 > 250 nM T92828 CE0L9G 10646375 IC50 > 2500 nM T92828 CSQR72 10646831 IC50 = 14000 nM T92828 C3U5HQ 10647021 IC50 = 18000 nM T92828 CKP13Z 10647488 IC50 > 100000 nM T92828 CG0H5R 10647642 IC50 > 2500 nM T92828 CGE27V 10647898 IC50 > 2500 nM T92828 C1TC3P 10648006 IC50 = 3500 nM T92828 C67RJH 10648135 IC50 = 67000 nM T92828 CYM2A6 10648715 IC50 = 35800 nM T92828 CKEB21 10648937 IC50 = 211 nM T92828 CC1G9O 10648996 Ki = 24.2 nM T92828 C6BNY8 10649086 IC50 = 1300 nM T92828 C34PRC 10649119 IC50 = 20 nM T92828 C2AN0W 10649321 IC50 = 960 nM T92828 CD6AP7 10649546 IC50 = 47800 nM T92828 C34WYT 10649585 IC50 = 50000 nM T92828 C32RCS 10650062 IC50 = 54000 nM T92828 CU25BJ 10650210 IC50 > 2500 nM T92828 C43LKS 10650331 IC50 > 100000 nM T92828 C5EG7D 10650477 IC50 = 6.9 nM T92828 CVJ6M3 10650546 IC50 = 600 nM T92828 CWH6N0 10651488 IC50 = 0.2 nM T92828 CQM4X9 10665805 IC50 = 15000 nM T92828 C17DRT 10669224 Ki = 34000 nM T92828 C7RE5Y 10670279 IC50 > 2500 nM T92828 CT50AW 10670372 IC50 = 5200 nM T92828 CQ7OS0 10670662 Ki = 1300 nM T92828 C0XV5H 10671031 Ki = 970 nM T92828 CRQ74D 10671036 IC50 > 2500 nM T92828 CCWP21 10671649 IC50 = 1500 nM T92828 CXT81R 10671928 IC50 = 3200 nM T92828 C85HCL 10672494 IC50 = 4370 nM T92828 C3W9OA 10673091 Ki = 94.1 nM T92828 C8VR3F 10673644 IC50 = 984 nM T92828 C1G6MP 10673715 IC50 = 34000 nM T92828 C24AKS 10673756 IC50 > 2500 nM T92828 CU36WQ 10673969 IC50 = 48000 nM T92828 CGV4O8 10674095 IC50 = 600 nM T92828 CKR7T8 10674176 IC50 = 445 nM T92828 CUOS92 10674642 IC50 = 44 nM T92828 CNQW61 10685758 IC50 > 100000 nM T92828 CK8O3S 10691437 Ki = 1700 nM T92828 CG6M7O 10692125 Ki = 3500 nM T92828 CPU9X8 10692351 IC50 > 2500 nM T92828 C0GPT3 10693110 IC50 > 2500 nM T92828 C2H8OE 10693607 Ki = 2500 nM T92828 C87FYW 10694591 IC50 = 11000 nM T92828 CWS8D4 10695071 IC50 = 9100 nM T92828 CS1IH0 10695363 IC50 > 2500 nM T92828 CCQ08V 10696210 IC50 = 32600 nM T92828 CW09TH 10696788 IC50 = 5900 nM T92828 CJN38O 10696818 IC50 = 72000 nM T92828 CH0K8I 10696876 IC50 > 100000 nM T92828 CC16FS 10697520 IC50 = 7.3 nM T92828 C28DBF 10697633 IC50 = 34000 nM T92828 CK61PF 10697636 IC50 = 29300 nM T92828 CW6K1Q 10697883 IC50 = 19800 nM T92828 C0YI4J 10698065 IC50 = 1.1 nM T92828 CN5X6J 10715441 IC50 = 29200 nM T92828 C2I8XQ 10717504 IC50 > 25000 nM T92828 CV64IK 10717923 IC50 = 8270 nM T92828 CG4JW8 10718141 IC50 > 2500 nM T92828 CAJV40 10718688 IC50 = 67500 nM T92828 CZJ4P6 10719007 IC50 = 27300 nM T92828 CHPV34 10719157 Ki = 1300 nM T92828 C43LWC 10719367 IC50 = 760 nM T92828 CQ6S3P 10719598 IC50 = 397 nM T92828 CAG5X7 10720982 IC50 = 2.1 nM T92828 C80JTH 10721484 Ki = 195 nM T92828 CQI32K 10722371 IC50 = 2300 nM T92828 C0K9DB 10722385 IC50 = 900 nM T92828 CCD61P 10722389 IC50 = 6.1 nM T92828 CZA8Y5 10723203 IC50 = 3.3 nM T92828 C6A5TD 10740258 Ki = 12000 nM T92828 CIO0Z4 10740439 IC50 = 44700 nM T92828 CT8L7G 10740614 IC50 = 18000 nM T92828 CC3OM9 10740953 Ki = 12000 nM T92828 CTC6N1 10741025 IC50 = 17700 nM T92828 CLT30A 10742005 Ki = 1800 nM T92828 C5J6YZ 10742841 IC50 > 2500 nM T92828 CGJ2T7 10742968 IC50 > 100000 nM T92828 C48MQX 10743346 Ki = 1400 nM T92828 CCA15K 10744040 IC50 = 81 nM T92828 CB74KC 10744085 IC50 = 2400 nM T92828 C1SAE7 10745418 IC50 = 26 nM T92828 CI5K1B 10745668 IC50 > 2500 nM T92828 C3EYA5 10746431 IC50 > 250 nM T92828 CPW0T6 10763862 Ki = 1100 nM T92828 CG7WB3 10765057 IC50 = 2000 nM T92828 C9WM1S 10765171 IC50 = 3900 nM T92828 CVOU41 10766198 IC50 = 97700 nM T92828 CCZA72 10766385 IC50 = 1410 nM T92828 C0BV7Q 10767280 IC50 = 36000 nM T92828 COUL31 10767505 IC50 = 3000 nM T92828 CFZ85A 10767778 IC50 = 2700 nM T92828 CPTF13 10768897 Ki = 14.7 nM T92828 CAEC98 10768903 IC50 = 5 nM T92828 CKWL78 10768904 IC50 = 3.4 nM T92828 C54XWU 10769177 IC50 = 3.8 nM T92828 CF0ZA8 10769526 IC50 = 1200 nM T92828 CULZ60 10769887 Ki = 40 nM T92828 CCN2M7 10786696 Ki = 160 nM T92828 CLR0N4 10788494 IC50 = 4800 nM T92828 CBW04Z 10788853 IC50 = 25000 nM T92828 CR93VH 10789524 IC50 = 260 nM T92828 C5KVM6 10789525 IC50 = 260 nM T92828 CIVE85 10790686 IC50 = 1600 nM T92828 C86RWA 10790757 IC50 = 950 nM T92828 C8W9ZS 10791694 IC50 = 2000 nM T92828 C4N1DZ 10791988 IC50 > 100000 nM T92828 C5Q9DW 10792316 IC50 = 20 nM T92828 C4IN2K 10792636 IC50 = 3.6 nM T92828 CL51IS 10792711 IC50 = 0.8 nM T92828 C69NMS 10792783 IC50 > 100000 nM T92828 C47DXJ 10792934 IC50 = 1.5 nM T92828 CBM8Y6 10793053 IC50 = 8.1 nM T92828 COUV95 10793160 Ki = 20 nM T92828 C8P1RH 10805820 IC50 > 100000 nM T92828 CKIV27 10811477 Ki = 94000 nM T92828 CD15AQ 10811595 IC50 = 14100 nM T92828 CCF2R5 10813228 Ki = 94000 nM T92828 CW4MP1 10814036 IC50 = 723 nM T92828 CAN8P9 10814297 Ki = 1500 nM T92828 C0LMU6 10814318 IC50 = 60000 nM T92828 CI9Y0N 10814440 IC50 = 1000 nM T92828 C3KS2I 10814743 IC50 = 2100 nM T92828 CO12UX 10814746 IC50 = 5500 nM T92828 CIF9U5 10814776 IC50 = 10100 nM T92828 C7AV5W 10815005 IC50 = 1900 nM T92828 CT2HR0 10815167 IC50 = 5890 nM T92828 C9LQ0A 10815168 IC50 = 6920 nM T92828 CT5C4K 10815239 Ki = 60 nM T92828 CQC01W 10815726 IC50 = 18 nM T92828 CQS3I2 10815823 IC50 = 240 nM T92828 CG7QW1 10816110 IC50 = 48000 nM T92828 CI98CT 10816152 IC50 = 57 nM T92828 CBG9H3 10816667 IC50 = 5 nM T92828 C7R4WU 10816682 IC50 > 2500 nM T92828 C6AKY9 10816963 IC50 = 0.85 nM T92828 C5B6SE 10817024 IC50 = 108 nM T92828 CF12ET 10818246 IC50 > 2500 nM T92828 C1UD8I 10832763 IC50 > 100000 nM T92828 C2TQO1 10833686 IC50 > 100000 nM T92828 C7OQ6G 10835335 Ki = 100000 nM T92828 CM40OP 10836754 Ki = 2500 nM T92828 COTE52 10837085 Ki = 6000 nM T92828 CWB28Y 10839533 IC50 = 37200 nM T92828 CB67FN 10839618 IC50 > 250 nM T92828 C80GEX 10839947 IC50 = 0.27 nM T92828 C1LD6J 10840410 IC50 = 4500 nM T92828 CO4WH7 10840560 Ki = 3.21 nM T92828 CC0OW9 10841170 IC50 = 1.1 nM T92828 CC3O7N 10841576 IC50 = 6.6 nM T92828 C8O0PJ 10854399 IC50 > 100000 nM T92828 CCP93B 10864118 Ki = 1700 nM T92828 CRFU13 10907333 Ki = 1100 nM T92828 CZ86ML 10918301 Ki = 150 nM T92828 CS08OB 10918368 Ki = 950 nM T92828 CCDS01 10918390 IC50 = 7700 nM T92828 C3ILH7 10929533 Ki = 550 nM T92828 CC3JY9 10941084 Ki = 320 nM T92828 CD85OB 10941181 Ki = 1400 nM T92828 CT1X9E 10972867 Ki = 4000 nM T92828 CME50A 10973161 Ki = 980 nM T92828 C5D3ZQ 10973218 Ki = 2700 nM T92828 C4P0HA 10983992 IC50 = 8130 nM T92828 C3RU0A 10984658 Ki = 1200 nM T92828 C50GTK 11006149 Ki = 2300 nM T92828 C3DJP1 11027595 Ki = 790 nM T92828 CY0R2V 11027946 IC50 = 950 nM T92828 C4QLF1 11038320 IC50 = 12000 nM T92828 CA26LW 11049336 Ki = 9100 nM T92828 C84YPI 11059912 Ki = 4800 nM T92828 CV1N7F 11071062 Ki > 50000 nM T92828 CV3EF2 11071347 IC50 = 1040 nM T92828 CA8C6B 11071765 Ki = 87 nM T92828 CFP0E7 11081276 Ki = 1700 nM T92828 CM51RW 11082049 Ki = 360 nM T92828 C4T1IB 11082168 Ki = 380 nM T92828 C4Q7VR 11103112 Ki = 4600 nM T92828 CT2X7H 11103181 Ki = 1300 nM T92828 CG8AD9 11103326 Ki = 1900 nM T92828 C91TLO 11113812 Ki = 1900 nM T92828 CTC76R 11123603 Ki = 4300 nM T92828 C3Q0LZ 11124425 Ki = 1500 nM T92828 CY9TE7 11124545 Ki = 2500 nM T92828 C0KC4B 11124821 Ki = 310 nM T92828 CN6R0S 11145758 Ki = 270 nM T92828 C2D5QN 11155687 IC50 = 87.8 nM T92828 C53FCK 11156301 IC50 = 261 nM T92828 C80CVQ 11156376 IC50 = 253 nM T92828 CTGR39 11156692 IC50 = 68.8 nM T92828 CP57YV 11157599 IC50 = 8620 nM T92828 C1X6ON 11167889 IC50 = 5600 nM T92828 C3ZJ8G 11168401 IC50 = 8030 nM T92828 C7VD8I 11168474 IC50 = 33.1 nM T92828 CPS0F6 11169125 IC50 = 109 nM T92828 CX9KE7 11191999 IC50 = 32.9 nM T92828 C90ZLV 11192437 IC50 > 1000 nM T92828 CN9VF3 11192438 IC50 > 1000 nM T92828 C36ZYQ 11192508 IC50 > 10000 nM T92828 CL5RD9 11202819 IC50 = 711 nM T92828 CUS0J1 11203972 IC50 > 10000 nM T92828 C07BRG 11204331 IC50 = 7.1 nM T92828 C6X3BJ 11224973 IC50 = 654 nM T92828 C3ZPJ8 11226740 IC50 = 184 nM T92828 CC23LY 11226767 IC50 = 966 nM T92828 CCV95P 11235126 IC50 = 3640 nM T92828 CG0W4N 11238500 IC50 = 78.2 nM T92828 CR9CW2 11238540 IC50 = 1470 nM T92828 CH6OD0 11273181 IC50 = 22.5 nM T92828 CZ3IE2 11283571 IC50 = 47.4 nM T92828 CB64EK 11284285 IC50 = 50.7 nM T92828 CX0IP1 11284400 IC50 > 10000 nM T92828 CS87FB 11307120 IC50 = 73.6 nM T92828 CLR79C 11307457 IC50 = 49.3 nM T92828 C1YK2H 11307805 IC50 = 25.5 nM T92828 CBEW43 11308052 IC50 = 33.2 nM T92828 CBC26X 11318409 IC50 = 16.7 nM T92828 C8YK9R 11318559 IC50 = 743 nM T92828 C18DIX 11318978 IC50 = 10.9 nM T92828 CAIG09 11330570 IC50 = 33.2 nM T92828 C2N3DR 11330923 IC50 = 13.6 nM T92828 CC35XI 11330927 IC50 = 392 nM T92828 C8SL3P 11331242 IC50 = 25 nM T92828 CW1OM0 11342005 IC50 = 25.3 nM T92828 C25GKE 11342089 IC50 = 94.3 nM T92828 CM5YT2 11353580 IC50 = 68 nM T92828 CS8H7Z 11362537 IC50 = 9250 nM T92828 C1BZ2Y 11364770 IC50 = 32.8 nM T92828 CC7X9Q 11365059 IC50 = 24.1 nM T92828 CA58FY 11375934 IC50 = 26.8 nM T92828 C1CZ8A 11376627 IC50 = 15.6 nM T92828 CC0L7O 11377200 IC50 = 89.8 nM T92828 CAN9R5 11385689 IC50 = 6270 nM T92828 CY0XU7 11386977 IC50 = 153 nM T92828 CZ7DR0 11387205 IC50 = 105 nM T92828 C5TES2 11387315 IC50 = 181 nM T92828 CY6IN3 11387934 IC50 = 86.8 nM T92828 C0K7AH 11397857 IC50 = 1810 nM T92828 CA2LW1 11398658 IC50 = 13.1 nM T92828 CH41WM 11398818 IC50 = 80.2 nM T92828 CI27JP 11408654 IC50 = 473 nM T92828 C8RPX0 11409474 IC50 = 39.9 nM T92828 CL3ZW6 11410074 IC50 = 18.3 nM T92828 C7H1JE 11410410 IC50 = 745 nM T92828 C3PDH6 11421392 IC50 = 18.5 nM T92828 CV62BJ 11421972 IC50 = 30.8 nM T92828 C7SJ6E 11432418 IC50 = 55 nM T92828 CLAI47 11432855 IC50 = 3530 nM T92828 CGY8F0 11441050 IC50 = 7840 nM T92828 C5HNO9 11444738 IC50 = 36.5 nM T92828 C7AY3C 11452452 IC50 > 10000 nM T92828 CZ47BI 11455999 IC50 = 3150 nM T92828 CR6SC4 11456110 IC50 = 74.9 nM T92828 C3RX2S 11465096 IC50 > 10000 nM T92828 CF6W3J 11467573 IC50 = 241 nM T92828 C61GUD 11477664 IC50 = 47.8 nM T92828 C0V6KP 11478553 IC50 = 72.7 nM T92828 CXSE25 11478911 IC50 = 28.8 nM T92828 CETK86 11488556 IC50 = 9480 nM T92828 C79SJN 11489174 IC50 = 82 nM T92828 CQM85J 11489318 IC50 = 21.5 nM T92828 CN4BV0 11489946 IC50 = 761 nM T92828 C2R3GN 11490160 IC50 = 534 nM T92828 CKZ29W 11505449 IC50 = 330 nM T92828 CQF3S5 11730445 Ki = 1400 nM T92828 CK9D4G 11731054 Ki = 640 nM T92828 CHU05Q 11733544 Ki = 7300 nM T92828 C9EF7M 11734435 Ki = 2800 nM T92828 C29SQH 11744509 IC50 > 2500 nM T92828 CPS5K7 11752174 IC50 = 1780 nM T92828 CX58WI 11753090 IC50 = 122 nM T92828 CLWM92 11753582 IC50 = 119 nM T92828 CTB8N9 11754273 Ki = 4400 nM T92828 C0ZQB3 11755275 IC50 = 200 nM T92828 CK0F7T 11757759 IC50 = 120 nM T92828 CIP68E 11762890 Ki = 1050 nM T92828 C8D6ZR 11785180 IC50 = 7780 nM T92828 CRLP96 11785813 IC50 = 49.7 nM T92828 CQE14M 11786120 IC50 = 3700 nM T92828 CFE86R 11794992 Ki = 20000 nM T92828 CQ7TL8 11797288 Ki = 1700 nM T92828 CTU41I 11797486 IC50 = 15700 nM T92828 CE9UG2 11798109 IC50 = 7590 nM T92828 C8FX7Z 11798228 IC50 > 25000 nM T92828 CUC28M 11798504 IC50 = 1080 nM T92828 CT6FQ7 11799503 IC50 = 47000 nM T92828 C07UEA 11799541 IC50 = 9080 nM T92828 C0CG3O 11799625 IC50 = 830 nM T92828 CJBD29 11799636 IC50 > 100000 nM T92828 C7Y5RM 11799973 Ki = 63 nM T92828 CREG48 11799974 Ki = 23.2 nM T92828 CK4ZF6 11800505 IC50 > 100000 nM T92828 CTH08J 11800649 Ki = 25.1 nM T92828 C9BF8Z 11800804 IC50 = 20000 nM T92828 CN4K1R 11801906 Ki = 130 nM T92828 CY0W8I 11812665 Ki = 11000 nM T92828 CQ8H3G 11813553 Ki = 580 nM T92828 C3U2GJ 11827489 IC50 = 3050 nM T92828 CJW2R5 11827657 IC50 = 300 nM T92828 C78LHI 12146375 IC50 > 100000 nM T92828 CS2Y5E 14041110 IC50 = 7900 nM T92828 CH95CP 14673588 IC50 > 100000 nM T92828 C7C5MB 15289330 IC50 = 210 nM T92828 CH68UI 15289331 IC50 = 7400 nM T92828 CTZ1E4 15342056 IC50 > 100000 nM T92828 CORE65 15410997 IC50 > 2500 nM T92828 C2QA8Y 15411002 IC50 > 2500 nM T92828 CC8BP3 15411003 IC50 > 2500 nM T92828 CC58ZF 15411005 IC50 = 1300 nM T92828 C2RNU5 15411009 IC50 = 2500 nM T92828 CGT4Q2 15453170 IC50 = 610 nM T92828 C1ROV7 15453172 IC50 = 140 nM T92828 CD7NK1 15453177 IC50 = 7900 nM T92828 CW0GJ1 15453178 IC50 = 13000 nM T92828 CJR1T8 15453179 IC50 = 1100 nM T92828 C58JIU 15453180 IC50 = 1200 nM T92828 CI63TE 15453209 IC50 = 46000 nM T92828 CGHV58 15453210 IC50 = 24000 nM T92828 C52HXB 18184179 IC50 = 3676 nM T92828 C8BGV5 18184194 IC50 = 24 nM T92828 CDU0W6 18184206 IC50 = 5402 nM T92828 C7D8KR 18184228 IC50 = 323 nM T92828 C6YPB0 18184229 IC50 = 84 nM T92828 CEO31D 18184234 IC50 = 103 nM T92828 C4MK2X 18184249 IC50 = 1537 nM T92828 CP3IL6 18184256 IC50 = 447 nM T92828 COB38T 18617284 IC50 = 7000 nM T92828 CG1TS0 18617288 IC50 = 20000 nM T92828 CBV58I 18617299 IC50 = 105000 nM T92828 C9PW8A 18617302 IC50 = 35000 nM T92828 C2PJ4H 18617303 IC50 = 13000 nM T92828 CI7W0J 18617314 IC50 = 14000 nM T92828 CO3F6N 18617318 IC50 = 39000 nM T92828 CNFU26 18617322 IC50 = 37000 nM T92828 CSP2T0 18617327 IC50 = 45000 nM T92828 C58ZQH 18617333 IC50 = 5300 nM T92828 CB9CL8 18617340 IC50 = 4700 nM T92828 C0LCU8 18617344 IC50 = 3800 nM T92828 CD7H9C 18617345 IC50 = 14000 nM T92828 CT8U7N 18617351 IC50 = 25000 nM T92828 CBS6A9 18617354 IC50 = 6700 nM T92828 CAP5D3 18617355 IC50 = 4000 nM T92828 C7VJ0E 18617363 IC50 = 24000 nM T92828 CE2NL8 18617366 IC50 = 3400 nM T92828 CC27DW 18617374 IC50 = 13000 nM T92828 C8V6XS 18617377 IC50 = 15000 nM T92828 C3JH0V 18617379 IC50 = 22000 nM T92828 C57JVD 18617381 IC50 = 74000 nM T92828 CBXP49 18617385 IC50 = 29000 nM T92828 CB42AR 18617389 IC50 = 13000 nM T92828 CFL1W8 18617393 IC50 = 17000 nM T92828 C6Q7CR 18617395 IC50 = 38000 nM T92828 C5OH8G 18617403 IC50 = 9400 nM T92828 CP0TM2 18617407 IC50 = 25000 nM T92828 C72QST 18660520 Ki = 22000 nM T92828 CLMZ12 18660521 Ki = 6300 nM T92828 C7R1HU 18660522 Ki = 130000 nM T92828 C2L4ID 18660523 Ki = 170000 nM T92828 CQ35FJ 18738878 IC50 = 68 nM T92828 CC23YB 18738879 IC50 = 69 nM T92828 CVMZ19 18738880 IC50 = 210 nM T92828 C0L6JX 18738881 IC50 = 1500 nM T92828 C0R6XF 18936171 IC50 = 2600 nM T92828 CVGX90 18936180 IC50 > 10000 nM T92828 CW5JB8 18995986 IC50 = 420 nM T92828 CKJ26Q 18995988 IC50 = 15000 nM T92828 C89KDZ 18995989 IC50 = 490 nM T92828 CUL4T0 18995990 IC50 = 29000 nM T92828 CZO82K 18995991 IC50 = 230 nM T92828 CZMR43 18995992 IC50 = 170 nM T92828 CSR67J 18995995 IC50 > 2500 nM T92828 C8CU9J 18995996 IC50 = 690 nM T92828 C24WKM 18995998 IC50 = 1100 nM T92828 CIY7D1 18995999 IC50 = 760 nM T92828 CG4T2P 18996000 IC50 = 6700 nM T92828 C41WAQ 19010490 IC50 = 1900 nM T92828 C8CPZ7 19010493 IC50 = 230 nM T92828 CFK4N3 19010508 IC50 = 1600 nM T92828 CGQL06 19085508 Ki = 48000 nM T92828 CJ4W8X 19085510 Ki = 20000 nM T92828 C5YOI3 19347988 IC50 > 25000 nM T92828 CE49LB 19385674 IC50 = 31000 nM T92828 CAH21E 19432649 IC50 = 70 nM T92828 CH9GX2 19432672 IC50 = 1240 nM T92828 C6OW3M 19735343 IC50 = 2000 nM T92828 C38JIZ 21041249 IC50 = 5208 nM T92828 CYNS68 21041264 IC50 = 158 nM T92828 C0EG5I 21041266 IC50 = 1474 nM T92828 C9WM5T 21041267 IC50 = 812 nM T92828 C6R5QB 21041273 IC50 = 516 nM T92828 CSU45B 21041278 IC50 = 82 nM T92828 CM56UH 21041283 IC50 = 210 nM T92828 C50SCK 21041284 IC50 = 63 nM T92828 CTH8F6 21041288 IC50 = 290 nM T92828 C5JIK7 21041297 IC50 = 686 nM T92828 CIVT14 21041307 IC50 = 555 nM T92828 CA5U7Z 21041324 IC50 = 784 nM T92828 CQ63RK 21041370 IC50 = 712 nM T92828 C91PNA 21041372 IC50 = 192 nM T92828 C2ASQ9 21462925 IC50 = 27 nM T92828 C5FBY0 21462927 IC50 = 200 nM T92828 CZB64L 21462932 IC50 = 120 nM T92828 C8QSU9 21979593 IC50 = 506 nM T92828 CB5KF0 21979601 IC50 = 525 nM T92828 CB7YS6 22009947 IC50 = 650 nM T92828 C6O5CM 22103385 Ki = 75000 nM T92828 C4FDK6 22103537 Ki = 39000 nM T92828 CQ2NK5 22103589 Ki = 150000 nM T92828 C02YLT 22103743 Ki = 52000 nM T92828 CLX1H5 22103787 Ki = 9400 nM T92828 C60JDI 22103797 Ki = 120000 nM T92828 C6G9YF 22467229 IC50 = 204 nM T92828 CSKR05 22467230 IC50 = 1140 nM T92828 CRZI09 22467234 IC50 = 906 nM T92828 CN21KV 22467235 IC50 = 34 nM T92828 CASM08 22467237 IC50 = 574 nM T92828 C21FKO 22467266 IC50 = 245 nM T92828 CHF5V9 22616255 IC50 = 30000 nM T92828 CA1RM2 22616257 IC50 = 27000 nM T92828 C0D9JA 22616258 IC50 = 26000 nM T92828 CV3O7Y 22616262 IC50 = 16000 nM T92828 CJTM39 22998396 IC50 = 74100 nM T92828 CI8EP7 22998414 IC50 = 48680 nM T92828 CV17XE 22998438 IC50 > 100000 nM T92828 CC4V5I 22998439 IC50 > 100000 nM T92828 C72NFC 22998446 IC50 = 2400 nM T92828 CR3HW0 22998447 IC50 = 35500 nM T92828 C15ZYN 22998456 IC50 = 335 nM T92828 CD91IN 22998508 IC50 = 95550 nM T92828 CD6SZ3 23288645 IC50 = 15 nM T92828 C3C4PE 23445219 IC50 = 56250 nM T92828 CIJ1C5 23445221 IC50 = 43200 nM T92828 C68XCT 23445224 IC50 > 100000 nM T92828 CA0G8O 23445227 IC50 = 5930 nM T92828 C6E2OR 23445241 IC50 > 100000 nM T92828 C4J7YM 23445250 IC50 = 1505 nM T92828 CTCP41 23445254 IC50 = 39770 nM T92828 CX95AD 23445256 IC50 = 9240 nM T92828 CGN9I1 23445272 IC50 = 9355 nM T92828 CEU2K7 23445284 IC50 = 28250 nM T92828 CJ9U1W 23445285 IC50 = 6106.7 nM T92828 C1QT2W 23445304 IC50 = 8895 nM T92828 C2EB0A 23445313 IC50 = 4280 nM T92828 CNJM59 23445317 IC50 > 100000 nM T92828 CG1P3S 23445325 IC50 > 100000 nM T92828 C68HIG 23445333 IC50 = 12450 nM T92828 CCMH86 23445336 IC50 = 1395 nM T92828 C9I3JT 23445345 IC50 > 100000 nM T92828 C4AG5C 23445354 IC50 = 43850 nM T92828 C4T5MS 23445358 IC50 = 21200 nM T92828 CCA74M 23445366 IC50 = 2450 nM T92828 C4Z1GC 23445379 IC50 = 4480 nM T92828 CN3G8K 23445388 IC50 = 64450 nM T92828 CSP3J7 23445404 IC50 = 9210 nM T92828 C5S0AP 23445408 IC50 = 2895 nM T92828 CCJ37R 23445410 IC50 > 100000 nM T92828 CGW8P2 23445412 IC50 = 68400 nM T92828 C7B6HX 23445421 IC50 = 4295 nM T92828 CZC52A 23445430 IC50 = 4130 nM T92828 CYF1C9 23445438 IC50 = 17850 nM T92828 C8AF2V 23445445 IC50 > 100000 nM T92828 C5WR4F 23445457 IC50 = 3070 nM T92828 CV1ER8 23445458 IC50 = 9955 nM T92828 CNM0T8 23445468 IC50 = 81400 nM T92828 C0VA4G 23445498 IC50 = 60300 nM T92828 CIC27H 23445505 IC50 > 100000 nM T92828 C17QTN 23445506 IC50 = 59100 nM T92828 CV1TW8 23445507 IC50 = 15600 nM T92828 C4D0BK 23445516 IC50 = 3275 nM T92828 C2G0WY 23445523 IC50 = 9550 nM T92828 C0VE5Q 23445533 IC50 = 3480 nM T92828 CIU74B 23445537 IC50 = 1305 nM T92828 CAM4F5 23445538 IC50 = 7275 nM T92828 C8S6HK 23445544 IC50 = 6635 nM T92828 C64LFR 23445547 IC50 = 13500 nM T92828 CV6ZO3 23445562 IC50 > 100000 nM T92828 C1CUD7 23445593 IC50 = 11700 nM T92828 CK28IV 23548251 IC50 > 10000 nM T92828 C7R6ZY 23548253 IC50 = 216 nM T92828 C6QBP1 23662235 IC50 = 8.3 nM T92828 CPH16E 23664197 IC50 = 38 nM T92828 CZP9W1 23665178 IC50 = 4550 nM T92828 CA50BD 23690609 IC50 = 1600 nM T92828 CG74JF 23705748 IC50 = 15700 nM T92828 CHQI17 23705749 IC50 = 1900 nM T92828 C32JUQ 24997097 IC50 = 15602.3 nM T92828 CW9D6N 25211074 IC50 = 2868.4 nM T92828 C7LI1Q 42630531 IC50 = 677 nM T92828 C8TE1M 42630532 IC50 = 1131.2 nM T92828 CW8MG1 42630654 IC50 = 1030 nM T92828 CL63TM 42630655 IC50 = 548.2 nM T92828 C05NBA 44177614 IC50 = 2085 nM T92828 CR8I5W 44211959 IC50 = 1200 nM T92828 CS6L8E 44212539 IC50 = 43 nM T92828 CXWM12 44213540 Ki = 30800 nM T92828 C7KP1R 44213959 IC50 = 60 nM T92828 CY6UZ1 44214320 IC50 = 219 nM T92828 CGP2D6 44215416 IC50 = 288 nM T92828 CU6GE5 44265871 Ki = 343 nM T92828 C6TNJ7 44266532 IC50 = 22000 nM T92828 C3B0YZ 44266537 IC50 = 4400 nM T92828 CQLH23 44266538 IC50 = 14500 nM T92828 CEN40G 44266540 IC50 > 25000 nM T92828 C3VGW6 44266542 IC50 = 2500 nM T92828 CVJ34I 44266549 IC50 = 3300 nM T92828 CTBY61 44266552 IC50 = 1100 nM T92828 CB8AT5 44266565 IC50 > 25000 nM T92828 C5L4PX 44266567 IC50 = 7000 nM T92828 CQX4I8 44266568 IC50 = 21000 nM T92828 CD3L0E 44266575 IC50 = 12000 nM T92828 CL6R1C 44266592 IC50 = 15000 nM T92828 C4KI0U 44266594 IC50 = 850 nM T92828 C3JPQ4 44266595 IC50 = 14000 nM T92828 CPU56S 44266621 IC50 > 25000 nM T92828 C9FZ2P 44266628 IC50 > 25000 nM T92828 C7UH4R 44266629 IC50 > 25000 nM T92828 CT7VN2 44266640 IC50 = 670 nM T92828 CTP3M2 44266645 IC50 > 25000 nM T92828 CDI8R1 44266646 IC50 = 1400 nM T92828 C6IW4B 44266649 IC50 > 25000 nM T92828 CN97HS 44266654 IC50 > 25000 nM T92828 CE8C3V 44266655 IC50 = 2400 nM T92828 CQ0G4Y 44266850 IC50 = 68 nM T92828 C4T2NO 44266881 IC50 = 8200 nM T92828 CNL7H5 44266886 IC50 = 130 nM T92828 C95YDQ 44266902 IC50 = 5100 nM T92828 CC5IY6 44266940 IC50 = 22000 nM T92828 C4K0DX 44267002 IC50 = 10000 nM T92828 C53IRS 44270498 IC50 = 90 nM T92828 CB5YF6 44270522 IC50 = 420 nM T92828 CXM1K7 44270523 IC50 = 1300 nM T92828 CV5SA1 44270524 IC50 = 800 nM T92828 CG5ZR9 44270602 IC50 = 540 nM T92828 C0WCV2 44274885 Ki = 4700 nM T92828 CJY0N4 44274960 Ki = 3000 nM T92828 CC0B8Z 44277840 Ki = 810 nM T92828 CJ9Q2O 44278003 IC50 = 870 nM T92828 C9PSJ0 44278161 IC50 = 1600 nM T92828 C7OHT4 44278215 IC50 = 420 nM T92828 C0GRH9 44278270 IC50 > 25000 nM T92828 C8UGF0 44279126 IC50 = 300 nM T92828 C8B5ID 44279127 IC50 = 230 nM T92828 C6BWO0 44279128 IC50 = 300 nM T92828 C2SQY1 44279129 IC50 = 2400 nM T92828 CA7CE3 44279309 IC50 = 190 nM T92828 CY7G4S 44279349 IC50 = 300 nM T92828 CD19IQ 44279350 IC50 = 1100 nM T92828 CMK16B 44279351 IC50 = 2400 nM T92828 CS94JH 44279370 IC50 = 280 nM T92828 CJ5KZ3 44279371 IC50 = 2100 nM T92828 C0HE1T 44279383 IC50 = 1000 nM T92828 CIU3Q9 44279413 IC50 = 890 nM T92828 CZ0J7H 44279439 IC50 = 4700 nM T92828 CP3D7U 44279677 IC50 = 1050 nM T92828 C04CFK 44283270 IC50 = 4 nM T92828 C1Z9MO 44283471 IC50 = 0.8 nM T92828 C8PY9L 44284041 IC50 = 78 nM T92828 CR8I5H 44284115 IC50 = 51 nM T92828 CRTC24 44284183 IC50 = 420 nM T92828 C0R8DG 44284184 IC50 = 45 nM T92828 C8DOW0 44284196 IC50 = 100 nM T92828 CG38VX 44284199 IC50 = 480 nM T92828 CHR04C 44284236 IC50 = 20 nM T92828 CPDN49 44284238 IC50 = 19 nM T92828 C12RKH 44284266 IC50 = 43 nM T92828 C16MGW 44284287 IC50 = 11 nM T92828 CB6IV3 44284288 IC50 = 43 nM T92828 CEJ9P3 44284292 IC50 = 14 nM T92828 CW2VK0 44284328 IC50 = 25 nM T92828 CQS3K4 44284329 IC50 = 88 nM T92828 CFSM06 44284381 IC50 = 290 nM T92828 CBP0H2 44284391 IC50 = 23 nM T92828 C02HIZ 44284405 IC50 = 25 nM T92828 C3PU2W 44284437 IC50 = 5.6 nM T92828 CJ04KH 44286764 Ki > 30000 nM T92828 C0UXK5 44291255 IC50 = 355500 nM T92828 C8LI6J 44291575 IC50 = 40400 nM T92828 CKON69 44291583 IC50 = 61000 nM T92828 C20VYP 44291584 IC50 > 100000 nM T92828 C3QT4K 44291602 IC50 > 100000 nM T92828 CC95RE 44291884 IC50 = 32600 nM T92828 C24SGF 44291897 IC50 = 12200 nM T92828 C74LWC 44298956 IC50 = 540 nM T92828 C8I9PO 44298982 IC50 = 300000 nM T92828 C0FNW3 44298988 IC50 = 500 nM T92828 CK6BU1 44299019 IC50 > 10000 nM T92828 CUTV49 44299020 IC50 > 10000 nM T92828 CLK7D3 44299023 IC50 = 1300 nM T92828 CS80KW 44304492 IC50 = 210 nM T92828 CU73DW 44307287 Ki = 4700 nM T92828 CWSO92 44307412 Ki = 3000 nM T92828 CU5VA9 44308286 IC50 > 100000 nM T92828 C9IDO6 44308287 IC50 > 100000 nM T92828 CZX62K 44308413 IC50 = 47000 nM T92828 CX8M3Q 44308414 IC50 = 30000 nM T92828 CLJT98 44308415 IC50 = 18000 nM T92828 C28YHW 44308426 IC50 > 100000 nM T92828 CA5WJ1 44308499 IC50 > 100000 nM T92828 CR8U1X 44309445 IC50 > 10000 nM T92828 C6UL9Q 44309488 IC50 = 5300 nM T92828 CY0P5V 44309814 IC50 = 330 nM T92828 CT36JL 44309897 IC50 = 440 nM T92828 CIM84F 44309996 IC50 = 300 nM T92828 CGO1R4 44310016 IC50 = 1600 nM T92828 CC3ZE2 44311135 IC50 = 120 nM T92828 CDSL53 44311218 IC50 = 2800 nM T92828 CSLX12 44311225 IC50 = 1000 nM T92828 CQJI05 44311232 IC50 = 49 nM T92828 C9KM0C 44311233 IC50 = 170 nM T92828 CR0E5T 44311283 IC50 = 144 nM T92828 COLR05 44311284 IC50 = 160 nM T92828 CW3M6Y 44311285 IC50 = 63 nM T92828 CBM46T 44311288 IC50 = 770 nM T92828 C01CDF 44311321 IC50 = 700 nM T92828 CLRE28 44311345 IC50 = 25 nM T92828 CN7C4F 44311346 IC50 = 14 nM T92828 CR06YA 44311516 IC50 = 19 nM T92828 CNR47S 44311527 IC50 = 200 nM T92828 CVI91E 44311528 IC50 = 60 nM T92828 CPT62F 44311692 Ki = 0.23 nM T92828 CL5KJ1 44311698 Ki = 4.4 nM T92828 C0GZL9 44311699 Ki = 0.76 nM T92828 CE5RU8 44311700 Ki = 0.23 nM T92828 C6COX5 44311701 Ki = 0.21 nM T92828 CC30ZG 44311726 Ki = 0.39 nM T92828 CB3G2V 44311727 Ki = 0.24 nM T92828 C9J6SX 44311728 Ki = 0.14 nM T92828 CIL3K7 44311763 Ki = 1.3 nM T92828 CUD78H 44311772 Ki = 0.49 nM T92828 CTCJ29 44311773 Ki = 0.7 nM T92828 C1YQW0 44311803 Ki = 0.23 nM T92828 CYV6P0 44311804 Ki = 0.24 nM T92828 C2ZN5I 44311805 Ki = 0.38 nM T92828 CEGV56 44311810 Ki = 24 nM T92828 C10LVB 44311838 Ki = 0.38 nM T92828 CD6AW7 44311849 Ki = 0.59 nM T92828 CF01CS 44311850 Ki = 0.5 nM T92828 C9B4XY 44311851 Ki = 0.79 nM T92828 CV1DH5 44311852 Ki = 0.6 nM T92828 C40EXJ 44311858 Ki = 3.2 nM T92828 CJD0Y3 44311873 Ki = 3.1 nM T92828 C45IUQ 44311915 Ki = 0.34 nM T92828 CXSC73 44311989 Ki = 3.5 nM T92828 CM4JA6 44312023 Ki = 1200 nM T92828 CB3YW0 44314173 IC50 = 29 nM T92828 CM2NJ4 44314579 IC50 = 5 nM T92828 C80SJM 44314619 IC50 = 1.1 nM T92828 CMNS53 44314802 IC50 = 130 nM T92828 C7AS9N 44314904 IC50 = 4 nM T92828 C1LU5S 44315008 IC50 = 3.6 nM T92828 CY36NW 44316458 IC50 = 33000 nM T92828 C39PCZ 44316515 IC50 = 20000 nM T92828 C4NZK2 44316526 IC50 = 59000 nM T92828 CYWQ80 44316527 IC50 = 58000 nM T92828 CUG3R0 44316768 IC50 = 23000 nM T92828 CV0FY7 44316831 IC50 = 27000 nM T92828 CM0X9O 44316973 IC50 = 49000 nM T92828 CNI1P7 44316993 IC50 = 90000 nM T92828 CKY04J 44317005 IC50 = 47000 nM T92828 C4ED2W 44317109 IC50 = 11000 nM T92828 CSO8W9 44317215 IC50 = 15000 nM T92828 CI7VO0 44322947 IC50 = 62050 nM T92828 CU3VH5 44327347 IC50 = 5900 nM T92828 CU3HD9 44327629 IC50 = 37 nM T92828 CF28EL 44327890 IC50 = 4400 nM T92828 CLKA68 44327903 IC50 = 900 nM T92828 CBZ3U7 44328087 IC50 > 1600 nM T92828 C4WS7B 44328089 IC50 = 1800 nM T92828 C6J3WT 44332735 IC50 > 2500 nM T92828 CL7P8D 44332842 IC50 > 2500 nM T92828 CIE78D 44333366 Ki = 71.2 nM T92828 CBRP45 44333578 IC50 = 87 nM T92828 CKC04D 44333598 IC50 = 65 nM T92828 C2BM9V 44333721 IC50 = 140 nM T92828 CU74CY 44333867 IC50 = 100 nM T92828 CL8Q2W 44333887 IC50 = 940 nM T92828 C48LXP 44333889 IC50 = 53 nM T92828 CS3HR9 44333913 IC50 = 30 nM T92828 C6BH7M 44334053 IC50 = 130 nM T92828 CNBR86 44334065 IC50 = 63 nM T92828 C0QDY5 44334084 IC50 = 530 nM T92828 C3QKF4 44334097 IC50 = 190 nM T92828 C7VSP8 44334128 IC50 = 14 nM T92828 CXR8T9 44334129 IC50 = 9.1 nM T92828 CK0C1Y 44334130 IC50 = 21 nM T92828 C0BX8D 44334145 IC50 = 14 nM T92828 C1I5CL 44334146 IC50 = 63 nM T92828 C4BJ7O 44334150 IC50 = 8.4 nM T92828 C1A2MU 44339655 IC50 = 39700 nM T92828 C1MVH8 44339662 IC50 = 29700 nM T92828 CV4R9Z 44339714 IC50 = 7000 nM T92828 CQ8R7S 44339755 IC50 > 100000 nM T92828 C8N7UJ 44339756 Ki > 4300 nM T92828 CWDY59 44339840 IC50 = 48000 nM T92828 C2H4FY 44340049 IC50 = 92700 nM T92828 CJRF02 44351961 IC50 = 1130 nM T92828 C7HM1L 44351968 IC50 = 1300 nM T92828 CPZ94S 44352026 IC50 = 14300 nM T92828 CBI32E 44352079 IC50 = 2140 nM T92828 CM37XP 44357035 IC50 > 100000 nM T92828 CHE24D 44357132 IC50 = 21000 nM T92828 C9U6VC 44357174 IC50 = 61000 nM T92828 CITF21 44357212 IC50 > 100000 nM T92828 CY69NR 44357391 IC50 = 55000 nM T92828 CUXG74 44365561 Ki = 20000 nM T92828 C3W9KH 44365878 Ki > 200000 nM T92828 C5JKC3 44371357 IC50 = 170 nM T92828 CXT37Q 44371394 IC50 > 10000 nM T92828 CO4TF3 44371396 IC50 = 6400 nM T92828 C6EPC3 44371410 IC50 = 300 nM T92828 CS2U0J 44371420 IC50 = 5200 nM T92828 CCD03X 44371421 IC50 = 2700 nM T92828 C92TXD 44371429 IC50 = 3500 nM T92828 C9XG7T 44371449 IC50 = 430 nM T92828 CK72FB 44371450 IC50 = 6800 nM T92828 CL7I9T 44371460 IC50 = 1900 nM T92828 CG4K8U 44371467 IC50 > 10000 nM T92828 CWNK92 44371495 IC50 = 13 nM T92828 CU2O5F 44371515 IC50 > 10000 nM T92828 C72FBI 44371516 IC50 = 1300 nM T92828 CK04MB 44371523 IC50 > 10000 nM T92828 C48HFY 44371531 IC50 = 660 nM T92828 C5BJ8H 44371532 IC50 = 1600 nM T92828 C4J1OD 44371571 IC50 = 3000 nM T92828 CKIA31 44371593 IC50 > 10000 nM T92828 C0F8EI 44371612 IC50 > 25000 nM T92828 CP3T7Z 44371671 IC50 = 14000 nM T92828 CE5V2B 44371773 IC50 = 8.6 nM T92828 CV5B9Z 44383535 IC50 > 25000 nM T92828 CZ07MY 44383536 IC50 = 148000 nM T92828 CTR86P 44383537 IC50 = 21000 nM T92828 CA7BX1 44383592 IC50 = 50000 nM T92828 CB2H4W 44383742 IC50 = 2970 nM T92828 CWC95L 44383753 IC50 = 2000 nM T92828 CYM1J5 44383754 IC50 = 2970 nM T92828 CC4EQ1 44384177 IC50 = 765 nM T92828 C5CK8M 44384557 IC50 > 10000 nM T92828 CS57OV 44384610 IC50 = 351 nM T92828 CX4B1W 44384611 IC50 = 258 nM T92828 CSY82J 44384651 IC50 = 3240 nM T92828 CK9W5F 44384652 IC50 = 4135 nM T92828 C4M7YA 44384656 IC50 = 5245 nM T92828 CQXM63 44384715 IC50 = 3169 nM T92828 C1N3SA 44384723 IC50 = 5660 nM T92828 CWQ32E 44384757 IC50 = 3280 nM T92828 CDM4X3 44384766 IC50 = 1950 nM T92828 C9ST7O 44384826 IC50 = 3330 nM T92828 C3ZO9F 44384852 IC50 = 295 nM T92828 C3IH2N 44384966 IC50 = 903 nM T92828 CSJ42C 44385008 IC50 = 100 nM T92828 CUF05M 44385127 IC50 = 5370 nM T92828 CJ02XC 44385162 IC50 > 1000 nM T92828 C43ADQ 44385412 IC50 = 2110 nM T92828 CSP1A8 44385522 IC50 = 873 nM T92828 C35IMP 44385523 IC50 = 299 nM T92828 C26DIF 44385576 IC50 = 746 nM T92828 C2E3SP 44385586 IC50 = 823 nM T92828 C4B8VR 44385792 IC50 = 8240 nM T92828 CG94RA 44385805 IC50 = 2620 nM T92828 CYV8Q4 44386002 IC50 = 4580 nM T92828 C6OYN9 44386069 IC50 = 420 nM T92828 CE42KT 44386161 IC50 = 2280 nM T92828 CADI16 44386162 IC50 = 2970 nM T92828 CI87SP 44386163 IC50 = 4670 nM T92828 C3X1MN 44386169 IC50 = 13 nM T92828 CEV6F7 44387124 IC50 = 5100 nM T92828 CK7XM9 44387128 IC50 = 300 nM T92828 CJ7Y4B 44387530 IC50 = 3.8 nM T92828 CXRQ21 44387531 IC50 = 7 nM T92828 C81XWQ 44387532 IC50 = 240 nM T92828 CW4SK9 44387533 Ki = 140 nM T92828 C5WBJ1 44387537 IC50 = 28 nM T92828 C6UFY8 44387538 IC50 = 220 nM T92828 CI8HL6 44404967 IC50 = 60 nM T92828 C0GO9C 44439102 IC50 = 6003 nM T92828 CIS54Q 44439103 IC50 = 1110 nM T92828 C97JIW 44439105 IC50 > 10000 nM T92828 CE6RC7 44439106 IC50 = 4690 nM T92828 CH7WG4 44439108 IC50 = 4510 nM T92828 C3E1GM 44439111 IC50 = 1910 nM T92828 C42LOW 44439114 IC50 = 4920 nM T92828 CD4NM1 44458399 IC50 = 450 nM T92828 C8LEA4 44458597 IC50 = 846 nM T92828 CBUI18 44458604 IC50 = 228 nM T92828 CR69LH 44458650 IC50 = 310 nM T92828 C5BEX8 44458669 IC50 = 1056 nM T92828 CV0S2K 44458670 IC50 = 94 nM T92828 CER1W7 44458999 IC50 = 1100 nM T92828 CAJY18 44459247 IC50 = 474 nM T92828 CPT5A8 44459272 IC50 = 2570 nM T92828 C37FQS 52943105 IC50 = 3119 nM T92828 C4YK3X 52944276 IC50 = 4387 nM T92828 C68GJL 52949155 IC50 = 713 nM T92828 CMLQ42 52949197 IC50 = 856 nM T92828 CD4GT1 52950137 IC50 = 1453 nM T92828 CP19OQ 53321140 IC50 = 31 nM T92828 CDB1Y8 56668902 IC50 > 100000 nM T92828 C8TSX9 58688005 IC50 = 203 nM T92828 CE97RP 58688006 IC50 = 611 nM T92828 C0IP5B 58688008 IC50 = 567 nM T92828 CU3B7D 67952994 IC50 = 461 nM T92828 CVO35E 70240112 IC50 = 29 nM T92828 C0VJ2M 71449713 IC50 = 2424 nM T92828 C49KEX 71451525 IC50 = 76 nM T92828 C7VJ0W 71451526 IC50 = 461 nM T92828 CR74NM 71451527 IC50 = 424 nM T92828 C1GA0F 71451528 IC50 = 552 nM T92828 CVA24Y 71451529 IC50 = 322 nM T92828 C2QI7H 71453356 IC50 = 468 nM T92828 CS79DP 71453357 IC50 = 19.3 nM T92828 CRD7T6 71455060 IC50 = 2829 nM T92828 C9JZM4 71455061 IC50 = 1765 nM T92828 CKL51C 71455062 IC50 = 145 nM T92828 CL4T8W 71455063 IC50 = 167 nM T92828 C4Q6LJ 71455064 IC50 = 457 nM T92828 CL76UZ 71455065 IC50 = 561 nM T92828 CB0EI6 71455139 IC50 = 5067 nM T92828 CUV4P7 71455140 IC50 = 2474 nM T92828 CYB60E 71456862 IC50 = 341 nM T92828 C7N3KS 71456863 IC50 = 147 nM T92828 C7LMX1 71456864 IC50 = 655 nM T92828 C3Q6IB 71456865 IC50 = 2490 nM T92828 C4XE8T 71456935 IC50 = 0.208 nM T92828 CP5OM0 71458717 IC50 = 9506 nM T92828 C5ZC7W 71458718 IC50 = 1501 nM T92828 CX2Q1M 71458719 IC50 = 42 nM T92828 CQ1C8Y 71458720 IC50 = 3479 nM T92828 CJ0ZG5 71458721 IC50 = 1082 nM T92828 C4H9GW 71460535 IC50 = 377 nM T92828 C3ZVU9 71460536 IC50 = 1146 nM T92828 C07SOZ 71460537 IC50 = 1474 nM T92828 CYS3W0 71460621 IC50 = 457 nM T92828 CA39BC 71462245 IC50 = 208 nM T92828 CX7C4B 71462246 IC50 = 194 nM T92828 CN3Z1G 71462247 IC50 = 166 nM T92828 CXG1J8 71462248 IC50 = 554 nM T92828 COUE65 71462320 IC50 = 441 nM T92828 CJCM28 71462321 IC50 = 1264 nM T92828 CA78CN 71462322 IC50 = 830 nM T92828 CHX9P8 71719083 IC50 = 29 nM T92828 C5GF1A 73345478 IC50 = 1.2 nM T92828 CD06SE 76308472 IC50 = 421 nM T92828 CVD37X 76312118 IC50 = 683 nM T92828 CS4AO6 76319370 IC50 = 240 nM T92828 C2G5FV 76330201 IC50 = 217 nM T92828 CEWB01 90663476 IC50 = 1.2 nM T92828 CWY29O 90766557 IC50 > 1000 nM T92828 C4DU0K 134131005 IC50 = 0.0063 nM T92828 CC1N3A 134157696 IC50 = 0.1 nM T92828 C1LD6M 135415889 IC50 = 2500 nM T92828 C8MXL7 135512539 IC50 = 294 nM T92828 C7O6VE 135884434 IC50 = 238 nM T92828 CN3ZE2 137633242 IC50 = 972 nM T92828 C23ACU 137633653 IC50 = 1435 nM T92828 C9IRL3 137637038 IC50 = 617.5 nM T92828 CX0YV5 137638953 IC50 = 758.3 nM T92828 C7IM5Q 137639474 IC50 = 1983 nM T92828 CDE50H 137642741 IC50 = 4072.1 nM T92828 C81EDX 137643691 IC50 = 935 nM T92828 CA60GK 137647152 IC50 = 698 nM T92828 CW34UP 137649592 IC50 = 803.2 nM T92828 CQ8Y5V 137649809 IC50 = 2156 nM T92828 C1EW4L 137651120 IC50 = 1.2 nM T92828 C09IFA 137652304 IC50 = 1353 nM T92828 C1WG3B 137655285 IC50 = 562 nM T92828 CRT9I5 137655525 IC50 = 16203.5 nM T92828 CD6W2K 137661460 IC50 = 1003.7 nM T92828 C1MI4T 155511294 IC50 = 3.5 nM T92828 C49YIT 155517241 IC50 = 315 nM T92828 C0YXP4 155519384 IC50 = 42 nM T92828 CO8N9V 155542285 IC50 = 90 nM T92828 CZN9I0 155544917 IC50 = 310 nM T92828 CW6FD5 155551580 IC50 = 120 nM T92828 CF6T1B 155560343 IC50 = 1.2 nM T92828 CJB9O1 155562688 IC50 = 1430 nM T92828 CPEX85 155563100 IC50 = 569 nM T92828 CGH80Y 155564169 IC50 = 542 nM T92828 D00RGL 44371672 IC50 = 15000 nM T92828 D06OSN 44371614 IC50 = 13000 nM T92828 D07OMS 9960931 IC50 = 1800 nM T92828 D0F6TS 16219332 IC50 = 0.0063 nM T92828 D0F8BZ 44371670 IC50 = 4300 nM T92828 D0G5UD 5312146 IC50 = 69 nM T92828 D0X1XM 9893800 Ki = 4.75 nM T92828 D0X1ZC 9848710 Ki = 36 nM T92828 D0Y1HN 5310991 IC50 = 6.4 nM T92828 D0Y8UY 44371613 IC50 = 7600 nM T14731 D06NVJ 936 IC50 < 50000 nM T14731 D0E3SH 6918837 Ki > 10000 nM T14731 D05KED 53340666 IC50 > 10000 nM T14731 D09XIZ 11538455 Ki > 10000 nM T14731 D0E3LP 5113032 IC50 = 85 nM T14731 D0H2UB 5361 IC50 = 300 nM T14731 D0M8FD 4261 IC50 > 100000 nM T14731 D0U3EP 445154 EC50 = 23600 nM T14731 D00RNS 49847188 IC50 > 90000 nM T14731 D04JZE 3246390 IC50 = 8850 nM T14731 D07NKC 49847118 IC50 = 39900 nM T14731 D0V2UZ 49847196 IC50 = 42700 nM T14731 CBY6Q1 2400 IC50 = 15700 nM T14731 CZQM89 7403 IC50 = 1000000 nM T14731 CZ25OS 8514 IC50 = 300 nM T14731 CJ7U9O 96455 IC50 = 17000 nM T14731 C3RUP6 443592 IC50 > 600000 nM T14731 C1C6RF 609412 IC50 > 100000 nM T14731 CH4L3B 626866 IC50 > 300000 nM T14731 CQ1MJ6 645092 IC50 > 300000 nM T14731 CY6L5C 648461 IC50 = 80000 nM T14731 C3OGK9 655862 IC50 = 22000 nM T14731 C01EIO 658354 IC50 > 300000 nM T14731 CLY6K3 661302 IC50 = 205 nM T14731 C6S1MX 661498 IC50 = 24800 nM T14731 C94MIR 662396 IC50 = 35600 nM T14731 C75SWH 662677 IC50 = 61300 nM T14731 CWM2C9 662768 IC50 = 88600 nM T14731 C5POL4 662842 IC50 = 19000 nM T14731 C36DRX 663194 IC50 = 20300 nM T14731 CVH0A6 665474 IC50 = 41000 nM T14731 C4EZF6 665718 Ki = 600 nM T14731 CEN23C 665743 IC50 = 29300 nM T14731 CFP62S 687118 Ki = 800 nM T14731 C9J6IC 694858 IC50 = 13000 nM T14731 C0J1SW 694859 IC50 = 12400 nM T14731 CBD84H 698853 IC50 = 10500 nM T14731 C7ZNC9 703333 IC50 = 29300 nM T14731 C8MBJ9 707029 IC50 = 160 nM T14731 CJ8L3N 707032 IC50 = 98 nM T14731 C5SMF6 746633 IC50 = 256000 nM T14731 CK0YJ1 787460 IC50 > 300000 nM T14731 C3V9CF 787462 IC50 > 300000 nM T14731 CT94VE 867287 IC50 > 300000 nM T14731 CTJA75 877268 IC50 = 243000 nM T14731 C29SYR 878744 IC50 > 300000 nM T14731 C5ITQ3 900927 IC50 = 240000 nM T14731 C50DGO 901929 IC50 = 56000 nM T14731 CT1J9H 914268 IC50 = 63 nM T14731 C5E9XG 914269 IC50 = 23000 nM T14731 C5RGM3 933903 IC50 = 27400 nM T14731 CGB37U 934700 IC50 = 7500 nM T14731 C1Y2TX 936014 IC50 = 31300 nM T14731 CS07QM 937168 IC50 = 27600 nM T14731 C1EZ5F 937643 IC50 = 46700 nM T14731 C5F7QG 1034419 IC50 > 100000 nM T14731 CW1L2Z 1068167 IC50 > 300000 nM T14731 C3VBZ9 1095092 IC50 = 3400 nM T14731 C0XD3L 1096276 IC50 > 100000 nM T14731 C1RVS5 1096292 IC50 > 50000 nM T14731 C6YS9Z 1103548 IC50 = 6700 nM T14731 C2Q1DX 1104317 IC50 = 9600 nM T14731 CGWC35 1114244 EC50 = 6000 nM T14731 CE4KD6 1142691 IC50 = 28400 nM T14731 CPI3Q1 1183101 IC50 > 50000 nM T14731 CU7ZT4 1183103 IC50 > 50000 nM T14731 CUJ7W0 1183104 IC50 > 50000 nM T14731 CLK57R 1183106 IC50 > 50000 nM T14731 CH9V7F 1183108 IC50 > 50000 nM T14731 CEP9Y7 1207797 IC50 = 198000 nM T14731 CG64LE 1208250 IC50 > 300000 nM T14731 CC54KV 1211361 IC50 = 146000 nM T14731 C5DIE4 1230959 IC50 = 424000 nM T14731 CWD2T7 1258010 IC50 = 6521000 nM T14731 CC8V0S 1328033 IC50 > 50000 nM T14731 CB7I9R 1372572 IC50 > 50000 nM T14731 CB92ZQ 1372991 IC50 = 9900 nM T14731 C4KIC0 1556677 IC50 > 40000 nM T14731 CW56UT 1736412 IC50 > 300000 nM T14731 C01HUX 1882365 EC50 < 1000 nM T14731 CG23UF 1915791 EC50 < 1000 nM T14731 C4JD2N 2130402 IC50 > 50000 nM T14731 CX8WT2 2248572 IC50 = 5300 nM T14731 C3ZS5K 2728632 IC50 = 78000 nM T14731 C0YS5J 2743189 IC50 = 192000 nM T14731 CDWU19 2827646 IC50 = 37000 nM T14731 CQ1T8A 2831741 IC50 > 100000 nM T14731 C3FJ9R 2834642 IC50 = 3100 nM T14731 CF2H5J 2848181 IC50 > 100000 nM T14731 CN6D2G 2858149 IC50 > 100000 nM T14731 CGN8J9 2859649 IC50 > 100000 nM T14731 CJG21Y 2915792 IC50 > 100000 nM T14731 CT1M7H 3106525 IC50 = 3466000 nM T14731 C50JXO 3130954 IC50 = 16350 nM T14731 C4OXA2 3148372 IC50 > 100000 nM T14731 CR3L5V 3163947 IC50 = 37900 nM T14731 C8VKW4 3163948 IC50 = 78000 nM T14731 CQFH65 3163949 IC50 = 76900 nM T14731 CLE4O2 3163950 IC50 = 4100 nM T14731 C9WT1X 3163951 IC50 = 47400 nM T14731 C2GQI5 3163952 IC50 = 51200 nM T14731 CL6S7W 3163955 IC50 = 20600 nM T14731 CP0WY4 3163956 IC50 = 45200 nM T14731 CJYP57 3163957 IC50 = 78800 nM T14731 CDE21Y 3163958 IC50 = 49800 nM T14731 C8TNV5 3163959 IC50 = 66600 nM T14731 C2TC1N 3205822 IC50 = 32000 nM T14731 CWB58P 3274235 EC50 < 1000 nM T14731 CGB17R 3290567 IC50 > 100000 nM T14731 CS0A8B 3459836 IC50 = 149 nM T14731 C94ELI 3610426 IC50 = 50500 nM T14731 CJ0T4E 3612016 IC50 = 180 nM T14731 CN8F1I 3953303 IC50 > 50000 nM T14731 CMJC34 4238838 IC50 = 110 nM T14731 CSO3R0 4893498 IC50 = 67000 nM T14731 CA83CZ 4893663 IC50 = 40700 nM T14731 C4U6VG 4893956 IC50 = 12200 nM T14731 CUCK41 4895138 IC50 = 8900 nM T14731 CE2HO8 4971057 IC50 = 48400 nM T14731 C35RHM 5811220 IC50 = 73000 nM T14731 CVC31J 6459022 IC50 = 110 nM T14731 C6JK5Y 6460292 IC50 = 18700 nM T14731 CD6VE3 6493840 IC50 = 23600 nM T14731 CO0ZW1 6493841 IC50 = 65700 nM T14731 CX3P2L 6493842 IC50 = 96200 nM T14731 CCY48M 6493843 IC50 = 75300 nM T14731 CGH01D 6493844 IC50 = 28700 nM T14731 C2CG9D 6493845 IC50 = 13700 nM T14731 C4BTL7 6493846 IC50 = 67900 nM T14731 C2LQT9 6493847 IC50 > 100000 nM T14731 CC8BK0 6496838 IC50 = 599000 nM T14731 CW14PR 6496840 IC50 = 1578000 nM T14731 CA5V1S 6918866 IC50 < 5000 nM T14731 CQ5NA2 7333748 IC50 = 36800 nM T14731 C2O4YS 9324490 IC50 = 783000 nM T14731 C7L2MG 10100985 IC50 = 9000 nM T14731 CON17T 10428959 IC50 = 34000 nM T14731 CY1JP2 11126879 IC50 = 21400 nM T14731 CT3WR4 11522166 IC50 > 100000 nM T14731 CYEK48 11536113 IC50 = 34500 nM T14731 C6TGJ1 11565551 IC50 = 2440 nM T14731 C7GA9I 11639738 IC50 > 200000 nM T14731 CC0VG2 11652227 IC50 = 79900 nM T14731 C6WMD3 11687587 IC50 = 77600 nM T14731 CQD76V 11694306 IC50 = 15000 nM T14731 CQ51EU 11701546 IC50 = 18000 nM T14731 CBYH25 11708252 IC50 = 2670 nM T14731 C63DRA 11708474 IC50 = 409 nM T14731 CXS96B 11840600 IC50 = 18800 nM T14731 CJ8L5T 11840601 IC50 = 29500 nM T14731 CYB16V 11854565 IC50 = 13000 nM T14731 CF7UG5 12476632 IC50 > 100000 nM T14731 C4DB8R 12761967 IC50 = 10500 nM T14731 CUS7H1 13505632 IC50 > 100000 nM T14731 CY1W2F 15701548 IC50 > 100000 nM T14731 CA4JG5 16805603 IC50 = 112000 nM T14731 CS31DN 21399939 IC50 = 2800 nM T14731 CHRA21 24168039 IC50 = 570000 nM T14731 CL2VP6 24180124 EC50 = 1800 nM T14731 CL4WV2 24180125 EC50 = 160 nM T14731 CQI29M 24180126 EC50 = 360 nM T14731 CI1R0Y 24772043 IC50 = 21000 nM T14731 CO6N3T 24822260 IC50 = 31000 nM T14731 CE73LG 24949066 IC50 = 325000 nM T14731 C9HJ0W 24949071 IC50 = 13000 nM T14731 CKN9H4 24949217 IC50 = 318000 nM T14731 CKRF97 24949372 IC50 = 168000 nM T14731 C4BL7A 25232161 EC50 = 130000 nM T14731 C37INZ 25232162 EC50 = 25000 nM T14731 C64BVL 25232163 EC50 = 31000 nM T14731 CU9K4V 25232345 EC50 = 990 nM T14731 C1O9DI 25232346 EC50 = 45000 nM T14731 CD06UK 25232347 EC50 = 610 nM T14731 C7XUO1 25233062 EC50 = 14000 nM T14731 CUE0K9 25233064 EC50 = 3700 nM T14731 CM1ZJ5 25233239 EC50 = 680 nM T14731 C73TAO 25233240 EC50 = 6900 nM T14731 CAH6Z1 25265679 EC50 < 250 nM T14731 CX96NF 42617956 IC50 = 12700 nM T14731 C9S7LC 42617959 IC50 = 43000 nM T14731 CAG4V5 42617960 IC50 = 44200 nM T14731 CFA67E 42617961 IC50 = 44500 nM T14731 C82LJW 42617968 IC50 = 50000 nM T14731 CPRD92 42617969 IC50 = 38300 nM T14731 CZ6H0F 42617970 IC50 > 90000 nM T14731 CI37UB 43358927 IC50 > 100000 nM T14731 CL0G4E 44138107 EC50 = 400 nM T14731 CCQ1R9 44138532 IC50 = 4000 nM T14731 CPV9R4 44405122 IC50 = 760 nM T14731 C9AX2Y 44427280 IC50 = 52000 nM T14731 CYL5A7 44565975 IC50 = 89800 nM T14731 CT5CK0 44572628 IC50 = 5000 nM T14731 C7OTS3 44572662 IC50 = 11100 nM T14731 CIP65R 44572663 IC50 = 4500 nM T14731 CR9C0G 44572664 IC50 = 12000 nM T14731 C89PGZ 44572666 IC50 = 310 nM T14731 CB9LM3 44572700 IC50 = 480 nM T14731 C1FXJ8 44572701 IC50 = 330 nM T14731 CV3JX8 44572702 IC50 = 570 nM T14731 CHE05V 44572703 IC50 = 4300 nM T14731 C9QF3T 44572704 IC50 = 180 nM T14731 C0OV2S 44572705 IC50 = 23200 nM T14731 C6NJG1 44572706 IC50 = 1400 nM T14731 C75FWN 44572767 IC50 = 230 nM T14731 CS0GP4 44572768 IC50 = 10800 nM T14731 CST4L3 44572769 IC50 = 3200 nM T14731 C4IF8W 44572770 IC50 = 220 nM T14731 C80SNU 44572771 IC50 = 6700 nM T14731 CC68AX 44572817 IC50 = 8800 nM T14731 C5EB9Z 44572818 IC50 = 380 nM T14731 CCRZ09 44572819 IC50 = 550 nM T14731 COYW18 44572820 IC50 = 180 nM T14731 C7M1DY 44572821 IC50 = 900 nM T14731 CQ2L0O 44591509 EC50 = 900 nM T14731 CK2EW9 44591510 EC50 = 4400 nM T14731 C1O0IE 44591533 EC50 = 300 nM T14731 C1IV3C 44591883 EC50 = 25000 nM T14731 CM86CB 44596232 IC50 = 52000 nM T14731 CRB83V 44596233 IC50 = 58000 nM T14731 C6L5KB 45168044 IC50 > 100000 nM T14731 CP06MS 45267617 IC50 = 89000 nM T14731 CU04RQ 45268494 IC50 = 68000 nM T14731 C2W8PE 45269359 IC50 = 60000 nM T14731 CL23BZ 45270178 IC50 = 58000 nM T14731 C50KMA 45270186 IC50 = 72000 nM T14731 C1FNP8 45272735 IC50 = 65000 nM T14731 C52OHP 45483031 IC50 = 9900 nM T14731 C67ICN 45486324 IC50 = 40000 nM T14731 CN14ZD 46226668 IC50 = 640 nM T14731 C28JLU 46226669 IC50 = 6000 nM T14731 CCEX52 46226675 IC50 = 34000 nM T14731 CW67RQ 46231289 IC50 = 8400 nM T14731 CSZ4B8 46856246 IC50 > 120000 nM T14731 CMF17W 46871954 IC50 = 2100 nM T14731 C4B0WG 46871955 IC50 = 5900 nM T14731 CND7M5 46919126 IC50 = 1800 nM T14731 CK4I9Y 46919223 IC50 = 223000 nM T14731 CBG93L 46966768 IC50 = 238000 nM T14731 C3ONP1 46966788 IC50 = 314000 nM T14731 CGD5W6 46966849 IC50 = 424000 nM T14731 C08ZDE 49806788 IC50 = 18300 nM T14731 C1KG4Q 49847039 IC50 > 90000 nM T14731 CG7JA8 49847120 IC50 = 46300 nM T14731 CH3L8A 49847124 IC50 > 90000 nM T14731 CIPU14 49847186 IC50 > 90000 nM T14731 CDXA49 49847190 IC50 > 90000 nM T14731 C1W9TL 49847192 IC50 > 90000 nM T14731 C3AVR6 49847270 IC50 = 36700 nM T14731 CVN51C 49847272 IC50 > 90000 nM T14731 CDM36I 49871498 IC50 = 37500 nM T14731 CLO50E 52941053 IC50 = 1767000 nM T14731 CPU09F 52941276 IC50 = 370 nM T14731 CMA1X5 52942684 IC50 = 11000 nM T14731 CQTG45 52943833 IC50 = 46000 nM T14731 C4GZ2T 52944947 IC50 = 122000 nM T14731 CO8TC4 52946220 IC50 = 40000 nM T14731 CDL1G9 52947355 IC50 = 240 nM T14731 CM4SC8 52947577 IC50 = 12000 nM T14731 CWS7J9 52947608 IC50 = 700 nM T14731 CBV42S 52947718 IC50 = 6100 nM T14731 C0UV1K 52948629 IC50 = 268000 nM T14731 C8QMO6 52949842 IC50 = 88000 nM T14731 C4JRF1 53257841 IC50 = 17500 nM T14731 CY4RF0 53258187 IC50 = 7700 nM T14731 CU64YT 53379498 IC50 = 89500 nM T14731 CV3B4K 54669816 IC50 = 1600 nM T14731 CXOK60 54669818 IC50 = 970 nM T14731 CLSD07 54669819 IC50 = 1300 nM T14731 CW3C4D 54757795 IC50 = 400 nM T14731 C3Z2WI 54757796 IC50 = 1000 nM T14731 CLOI75 54757797 IC50 = 660 nM T14731 CH18SI 54757799 IC50 = 51000 nM T14731 CE1X5Z 54757800 IC50 = 370 nM T14731 C8G7SA 54757892 IC50 = 770 nM T14731 CG19XC 54757893 IC50 = 18000 nM T14731 C1VJ5D 54757894 IC50 = 990 nM T14731 CQ95SY 54757895 IC50 = 1300 nM T14731 C62TLD 54757896 IC50 = 1000 nM T14731 C8SFD1 54757989 IC50 = 23000 nM T14731 CV6J3B 54757990 IC50 = 7400 nM T14731 CDI95E 54757991 IC50 = 5100 nM T14731 CPFX20 56663060 IC50 = 98 nM T14731 C3T8YQ 56664966 IC50 = 290000 nM T14731 CKFY59 56669934 IC50 = 12400 nM T14731 CC7T2A 56674921 IC50 = 41600 nM T14731 C6ZD1F 56676724 IC50 > 100000 nM T14731 CZ25SN 56935695 IC50 > 100000 nM T14731 C71BDL 57345649 IC50 = 21700 nM T14731 C32DTV 57391608 IC50 = 35800 nM T14731 C03DKB 57392691 IC50 > 90000 nM T14731 CV84RT 57395072 IC50 = 16100 nM T14731 CVDK34 57395074 IC50 > 60000 nM T14731 CCMV32 57398538 IC50 = 70900 nM T14731 C5FR8C 57398601 IC50 = 24700 nM T14731 CA9NY1 57400270 IC50 = 60200 nM T14731 CH0FE1 57403131 IC50 = 17900 nM T14731 C78NLU 58101565 EC50 < 250 nM T14731 CJ09SD 58101566 EC50 < 250 nM T14731 C92ZDR 59053311 IC50 > 2000 nM T14731 CE4IP3 60141294 IC50 = 6200 nM T14731 CM08ZL 60148504 IC50 > 100000 nM T14731 CV8E9Z 60150563 IC50 = 11080 nM T14731 C47BFO 60150564 IC50 = 43140 nM T14731 C5V3GZ 60150584 IC50 = 10130 nM T14731 C1CYX6 60150585 IC50 = 43290 nM T14731 CX57EP 60165377 IC50 > 100000 nM T14731 C02PIZ 60165378 IC50 > 100000 nM T14731 CV7JQ9 60165379 IC50 > 100000 nM T14731 C98IZK 60165380 IC50 = 210000 nM T14731 CE81YX 60165381 IC50 > 300000 nM T14731 CT1SK2 60165382 IC50 > 300000 nM T14731 C25HQM 60165383 IC50 > 300000 nM T14731 C4D6HC 60165506 IC50 > 100000 nM T14731 CA19BZ 60165642 IC50 > 100000 nM T14731 CV1YC9 60165643 IC50 > 100000 nM T14731 C9HR5A 60165644 IC50 > 100000 nM T14731 C70XDP 60165645 IC50 > 100000 nM T14731 C4AV6N 60165646 IC50 > 100000 nM T14731 CE89WD 60165647 IC50 > 100000 nM T14731 CSVW05 60165648 IC50 > 100000 nM T14731 CZ8NB6 60165794 IC50 > 100000 nM T14731 CCIV73 60165795 IC50 > 100000 nM T14731 CBY8D0 60165796 IC50 > 100000 nM T14731 CTRX85 60165797 IC50 > 100000 nM T14731 C2BN5H 60165798 IC50 > 100000 nM T14731 CH10ND 60165799 IC50 > 100000 nM T14731 CBWX25 60167125 IC50 > 100000 nM T14731 C1I3MW 60167126 IC50 > 100000 nM T14731 COH2I7 60167127 IC50 > 100000 nM T14731 C6SWQ8 60167128 IC50 > 100000 nM T14731 CR3IQ7 60167129 IC50 > 100000 nM T14731 C0TO6E 60167270 IC50 > 100000 nM T14731 C43YCN 60167271 IC50 > 100000 nM T14731 C3HCS6 60167272 IC50 > 100000 nM T14731 CI9DZ5 60167273 IC50 > 100000 nM T14731 C04PIO 60167274 IC50 > 100000 nM T14731 C92UWL 60167276 IC50 > 100000 nM T14731 C5JGZ2 60167277 IC50 > 100000 nM T14731 CJ8MU4 60167418 IC50 > 100000 nM T14731 C8DA7M 60167419 IC50 > 100000 nM T14731 CCI6D7 60167420 IC50 > 100000 nM T14731 CAMB94 60167421 IC50 > 100000 nM T14731 C53FNR 60167422 IC50 > 100000 nM T14731 C4G6LE 60167423 IC50 > 100000 nM T14731 COHB83 60167424 IC50 > 100000 nM T14731 C94IGH 66560391 IC50 > 200000 nM T14731 CWM6Z8 67523832 IC50 = 75000 nM T14731 C0Q6FC 68509298 IC50 > 100000 nM T14731 C0LV7N 70089831 IC50 > 100000 nM T14731 C78HWC 70676483 IC50 = 7000 nM T14731 CL2J4U 70676484 IC50 = 20200 nM T14731 CDO4B9 70676622 IC50 = 9400 nM T14731 C5Y0CD 70676623 IC50 = 6600 nM T14731 C9ZA7E 70676624 IC50 = 10400 nM T14731 CSZ76Q 70676625 IC50 = 21100 nM T14731 C3DHW2 70676626 IC50 = 12000 nM T14731 CE80CA 70676627 IC50 = 11800 nM T14731 CA4PI8 70676628 IC50 = 12500 nM T14731 CJ3SZ9 70676792 IC50 = 14100 nM T14731 C3X1ON 70685393 IC50 = 40060 nM T14731 CB15VL 70685403 IC50 = 25018 nM T14731 C57UAH 70691733 IC50 = 45970 nM T14731 CNVG06 71304813 IC50 = 3.6 nM T14731 CWY4S0 71304814 IC50 = 15 nM T14731 C4BHW5 71304815 IC50 = 4.3 nM T14731 CB4A3W 71451254 IC50 > 100000 nM T14731 C7LB1U 71451255 IC50 = 93000 nM T14731 CG1EW3 71451256 IC50 > 100000 nM T14731 C9N8WG 71451257 IC50 > 100000 nM T14731 C8CLX3 71452171 IC50 = 56500 nM T14731 CY0WC4 71453621 IC50 = 1000 nM T14731 C73LSH 71453984 IC50 = 53200 nM T14731 C43MRT 71455173 EC50 < 1000 nM T14731 CRF65P 71458450 IC50 > 100000 nM T14731 CF1W7G 71458835 IC50 = 43000 nM T14731 C1O0HF 71459392 IC50 = 6000 nM T14731 C31MUQ 71654770 IC50 > 50000 nM T14731 CU31DP 71654771 IC50 = 6.7 nM T14731 CAM70V 71654772 IC50 = 14 nM T14731 CE73FM 71654773 IC50 = 5.8 nM T14731 COV26M 71654774 IC50 = 110 nM T14731 CQ1KA4 71654775 IC50 = 15000 nM T14731 CMR87Y 71654838 IC50 > 50000 nM T14731 CAD5K9 71654839 IC50 = 16000 nM T14731 CTF4Y0 71654840 IC50 = 1600 nM T14731 CU46KD 71654841 IC50 = 56 nM T14731 C4RA6P 71654842 IC50 = 490 nM T14731 C3WYU5 71654843 IC50 = 4300 nM T14731 C12RAH 71654909 IC50 = 42 nM T14731 COW48U 71654910 IC50 = 120 nM T14731 C4AP1G 71654911 IC50 = 380 nM T14731 C1O0ZQ 71654912 IC50 = 730 nM T14731 CC6AJ7 71654913 IC50 = 110 nM T14731 CUHV94 71654914 IC50 = 53 nM T14731 CA2EM4 71654987 IC50 = 470 nM T14731 CNU2D1 71654988 IC50 = 59 nM T14731 CU5HD4 71654989 IC50 = 490 nM T14731 CP71AF 71654990 IC50 = 180 nM T14731 CUE91W 71654991 IC50 > 50000 nM T14731 CQOW51 71654992 IC50 > 50000 nM T14731 CS0FQ4 71654993 IC50 > 50000 nM T14731 CLDB05 71655060 IC50 = 5.3 nM T14731 C6JCD7 71655061 IC50 = 67 nM T14731 CX85ID 71655062 IC50 = 31 nM T14731 C8TX2W 71655063 IC50 = 17 nM T14731 C1TC4J 71655141 IC50 = 1600 nM T14731 C3CI5Q 71717360 IC50 = 31200 nM T14731 CM2J1S 71717361 IC50 = 88000 nM T14731 CC4Y0R 71717955 IC50 = 41700 nM T14731 CT8L3F 71718571 IC50 = 71400 nM T14731 CJ6IA8 71718835 EC50 = 1700 nM T14731 CG8UI2 71719783 IC50 = 45100 nM T14731 CEIX13 71812123 IC50 = 28000 nM T14731 CB5R9X 72550523 IC50 = 26000 nM T14731 CZ57NL 72550525 IC50 = 21000 nM T14731 CQ7M9B 72550526 IC50 > 100000 nM T14731 C2MFT3 72550527 IC50 = 38000 nM T14731 CU0WX7 72550747 IC50 > 250000 nM T14731 CKMS38 72550748 IC50 = 16700 nM T14731 C2R4FH 72664790 IC50 = 121200 nM T14731 CK6JB1 72664791 IC50 = 32100 nM T14731 CYZ9R7 72664892 IC50 > 200000 nM T14731 C6EFG7 73291970 IC50 = 240 nM T14731 CMS0F6 73292335 IC50 = 890 nM T14731 CMY90N 73292338 IC50 = 5980 nM T14731 C24SZG 73333807 IC50 = 58430 nM T14731 CD41CU 73333808 IC50 = 74520 nM T14731 CT3XY9 73333924 IC50 = 80110 nM T14731 CPLI82 73355035 IC50 = 297 nM T14731 CRZ62F 73355036 IC50 = 6700 nM T14731 C87LDV 77461130 IC50 > 100000 nM T14731 C67MJT 77461131 IC50 > 100000 nM T14731 C6LE9I 90016528 IC50 = 20000 nM T14731 C8XVT3 90645142 IC50 = 60310 nM T14731 CH1RY4 90645143 IC50 = 49120 nM T14731 CZIX41 90645144 IC50 = 79870 nM T14731 C9YIS4 90654860 IC50 = 41000 nM T14731 C76QJZ 90654861 IC50 = 37000 nM T14731 CAD9C4 90654862 IC50 = 26000 nM T14731 C9U5QY 90654863 IC50 = 21000 nM T14731 CG6Z9E 90654864 IC50 > 200000 nM T14731 CM3Q9R 90665503 Ki = 2600 nM T14731 CW0KC2 90665505 IC50 > 1000000 nM T14731 CUX71H 90666423 IC50 > 120000 nM T14731 C3FY9T 90666424 IC50 = 61900 nM T14731 CCKT95 90666431 IC50 = 58200 nM T14731 CZ6CX5 90666432 IC50 > 120000 nM T14731 CRH54C 90666436 IC50 = 68100 nM T14731 CL3TK7 90666629 IC50 = 4200 nM T14731 C0AMP1 90666630 IC50 = 3500 nM T14731 C8NO1T 90666631 IC50 = 6000 nM T14731 CU08OF 90666632 IC50 = 4100 nM T14731 C9YA6W 90666633 IC50 = 700 nM T14731 CV8JY4 90667869 IC50 = 2000 nM T14731 C5US4A 91673681 IC50 = 33600 nM T14731 CQO1F3 91673682 IC50 > 50000 nM T14731 C03GAW 98185391 IC50 = 7000 nM T14731 CP43XT 101884802 IC50 = 18700 nM T14731 CSDE45 101884803 IC50 = 64000 nM T14731 CW3TR5 101884804 IC50 = 22400 nM T14731 C48DRM 101884805 IC50 = 3820 nM T14731 CKR05E 101884807 IC50 = 11700 nM T14731 CM40UV 101884808 IC50 = 12000 nM T14731 CA15KO 101884809 IC50 = 788 nM T14731 CBJ50G 101884810 IC50 = 30300 nM T14731 CA7MT5 101884812 IC50 = 100000 nM T14731 C0W1CO 101884813 IC50 = 33600 nM T14731 CH06TS 101884814 IC50 = 13500 nM T14731 C2QJB4 101884815 IC50 = 4890 nM T14731 CZ17MX 101884816 IC50 = 40900 nM T14731 C2VX8K 112499922 IC50 > 100000 nM T14731 CM48HY 118283202 IC50 = 63000 nM T14731 CY2SJ0 118283203 IC50 > 100000 nM T14731 CHR58E 118283204 IC50 > 100000 nM T14731 C0Y8BI 118283209 IC50 = 56000 nM T14731 CL3X7K 118717122 IC50 = 26900 nM T14731 CY05KA 118717208 IC50 = 15400 nM T14731 CZQB67 118717209 IC50 = 70700 nM T14731 CZ5CB6 118718013 IC50 = 9000 nM T14731 CCLI64 118722847 IC50 > 100000 nM T14731 C9PF2T 118738000 IC50 = 1000 nM T14731 C1T6WZ 118738004 IC50 = 1200 nM T14731 CEJ3I2 118738006 IC50 = 2600 nM T14731 C7JWC8 118738008 IC50 = 1900 nM T14731 CI4M8F 118738010 IC50 = 6200 nM T14731 CNHA13 118738014 IC50 = 11000 nM T14731 CKO2H0 118738015 IC50 = 1700 nM T14731 CC3W5X 118738016 IC50 = 3100 nM T14731 CD71WH 118738018 IC50 = 2700 nM T14731 CAV76G 118738024 IC50 = 2100 nM T14731 CI2LJ9 118738026 IC50 = 800 nM T14731 CQM08D 121231415 Ki = 5000 nM T14731 C0D2KV 121313586 IC50 = 119400 nM T14731 CP8TX5 122180739 IC50 = 35250 nM T14731 CT9O7E 122180740 IC50 = 37360 nM T14731 CG6FI5 122184875 IC50 = 49900 nM T14731 C1K9SO 122184876 IC50 = 5600 nM T14731 C1QIE4 122184877 IC50 = 83400 nM T14731 CYLF42 122184878 IC50 = 117900 nM T14731 CA6R4T 122184879 IC50 = 62900 nM T14731 CR86MS 122184881 IC50 > 100000 nM T14731 CVM95G 122186869 IC50 = 630 nM T14731 C5ZYP0 122186870 IC50 = 2850 nM T14731 C97VZS 122186871 IC50 = 1960 nM T14731 CP5R3G 122186872 IC50 = 1150 nM T14731 CEOS03 122186873 IC50 = 1450 nM T14731 C95ZQN 122186874 IC50 = 640 nM T14731 CLO15R 122186875 IC50 = 2400 nM T14731 CML8G1 122186876 IC50 = 18900 nM T14731 C41TOB 122186877 IC50 = 6600 nM T14731 C57FWN 122186878 IC50 = 6600 nM T14731 CESR15 122186879 IC50 = 9600 nM T14731 C02XHR 122187733 IC50 = 6860 nM T14731 C5MGT9 122187734 IC50 = 2780 nM T14731 C5XE4R 122187735 IC50 = 10710 nM T14731 CNIL28 122187736 IC50 = 2130 nM T14731 C9KT4V 122187737 IC50 = 14430 nM T14731 CBAG46 122187738 IC50 = 3650 nM T14731 CSU7W2 122187739 IC50 = 12570 nM T14731 C9J3MI 122187740 IC50 = 3030 nM T14731 C2NEW8 122187741 IC50 = 2320 nM T14731 CVX6G1 124155856 IC50 = 12500 nM T14731 C8R1KL 124155864 IC50 = 6320 nM T14731 CKU31X 124155865 IC50 = 11300 nM T14731 C1VNS9 124155880 IC50 = 30200 nM T14731 CI5SG4 124155887 IC50 = 15600 nM T14731 C8D6VI 124155892 IC50 = 31400 nM T14731 CE9HV7 124155894 IC50 = 71500 nM T14731 CL43GB 124155906 IC50 = 14900 nM T14731 C98FJW 124155909 IC50 = 2230 nM T14731 CG4KQ0 124155918 IC50 = 2270 nM T14731 C2SK7Z 124155921 IC50 = 483 nM T14731 CI3K8Z 124155944 IC50 = 7920 nM T14731 CC6E5F 124155947 IC50 = 1620 nM T14731 CDK5F1 124156051 IC50 = 4190 nM T14731 C5H1WI 124156054 IC50 = 50800 nM T14731 CK10FP 124156076 IC50 = 7140 nM T14731 CZ1X0F 124156082 IC50 = 8020 nM T14731 CN6YV0 124156084 IC50 = 367 nM T14731 C6VX3U 124156175 IC50 = 237 nM T14731 CA47GR 124156294 IC50 = 10500 nM T14731 C94NWB 124156297 IC50 = 8540 nM T14731 CLU7F3 124156311 IC50 > 200000 nM T14731 C25ACW 124156314 IC50 = 5660 nM T14731 CC3H9B 124156319 IC50 = 3030 nM T14731 C0F8RC 124156322 IC50 = 3470 nM T14731 CH2BJ7 124156324 IC50 = 2460 nM T14731 CC1B5Q 124156332 IC50 = 24100 nM T14731 CZ43QA 124156333 IC50 = 13500 nM T14731 CWT8L7 124156337 IC50 = 8090 nM T14731 C2CIJ9 124156338 IC50 = 42400 nM T14731 CU51OV 124156339 IC50 > 200000 nM T14731 CM64KZ 124156375 IC50 = 2820 nM T14731 CS8D4J 124156389 IC50 = 145000 nM T14731 CO71HP 124156406 IC50 = 15300 nM T14731 CTF86E 124156432 IC50 = 10100 nM T14731 CH2MQ3 124156454 IC50 = 13400 nM T14731 C5A1MN 124156461 IC50 = 33300 nM T14731 C4DR7M 124156464 IC50 = 1550 nM T14731 C6Z3EX 124156466 IC50 = 30400 nM T14731 CQ1D7V 124156477 IC50 = 6270 nM T14731 CVG8H3 124156515 IC50 = 7330 nM T14731 CB6WM9 124156519 IC50 = 7970 nM T14731 C5X2EL 124156548 IC50 = 15500 nM T14731 COW18T 124156563 IC50 = 52100 nM T14731 C3R8OJ 124156568 IC50 = 18800 nM T14731 CJ2F5B 124156573 IC50 = 21000 nM T14731 CJ4C0I 124156580 IC50 = 142000 nM T14731 CF06XJ 124156582 IC50 = 9500 nM T14731 CJQC71 124156591 IC50 = 192000 nM T14731 C47GML 124156596 IC50 = 11300 nM T14731 CUJ71O 124156601 IC50 = 974 nM T14731 CK74XR 124156666 IC50 = 115000 nM T14731 CD83AZ 124156671 IC50 = 1230 nM T14731 COD08A 124156677 IC50 = 65200 nM T14731 C0R9GV 124156702 IC50 = 44600 nM T14731 CNT71Z 124156707 IC50 = 672 nM T14731 C7I1AZ 124156715 IC50 = 19700 nM T14731 CZDJ49 124156728 IC50 = 18700 nM T14731 CE1J6Y 124156731 IC50 = 2550 nM T14731 COTD57 124156742 IC50 = 1810 nM T14731 CLA01I 124156756 IC50 > 200000 nM T14731 CP36XI 124156875 IC50 = 9930 nM T14731 C9KP4E 124156885 IC50 = 90900 nM T14731 CSM9Q8 124156886 IC50 = 14700 nM T14731 C2CI9E 124156887 IC50 = 48500 nM T14731 CUBJ73 124156888 IC50 = 2230 nM T14731 CV1R2F 124156892 IC50 = 3010 nM T14731 CULA86 124156896 IC50 > 200000 nM T14731 CFN1X9 124156913 IC50 = 1880 nM T14731 CH9R8A 124156914 IC50 = 11500 nM T14731 C4AXU0 124156920 IC50 = 21800 nM T14731 C4Y8GT 124156967 IC50 = 20300 nM T14731 C2DKH0 124157048 IC50 = 192000 nM T14731 C4G2NW 124157054 Ki > 100000 nM T14731 CDR98I 124162056 IC50 = 3510 nM T14731 CJ47PM 126720627 IC50 = 42900 nM T14731 CU4IC8 126843233 IC50 = 98000 nM T14731 CU02IS 127027826 IC50 > 100000 nM T14731 C3DVH2 127028117 IC50 > 100000 nM T14731 CX9S6O 127032844 IC50 = 47 nM T14731 C8CV4N 127033814 IC50 = 165.1 nM T14731 C4J8WR 127034092 IC50 = 37.1 nM T14731 CH02OR 127034093 IC50 = 56.8 nM T14731 CJO78L 127034094 IC50 = 38.7 nM T14731 CY8TS5 127034095 IC50 = 2.3 nM T14731 C6FGW5 127034098 IC50 = 75.2 nM T14731 CCEP75 127034360 IC50 = 63.5 nM T14731 CZ2R6J 127035147 IC50 = 57500 nM T14731 CXR74F 127035863 IC50 = 62900 nM T14731 CB0K5D 127042242 IC50 = 3930 nM T14731 C3MP0W 127045459 IC50 = 9000 nM T14731 C84XPC 127048873 IC50 = 2080 nM T14731 CBJD15 127049868 IC50 = 1390 nM T14731 C7P8JZ 129883511 IC50 > 50000 nM T14731 CZ45LV 129906245 IC50 > 50000 nM T14731 CCH2T8 129906312 IC50 = 7700 nM T14731 C6X3HG 132145728 IC50 > 20000 nM T14731 C8O9DP 132157820 IC50 > 20000 nM T14731 CY8B2P 132837649 IC50 = 10220 nM T14731 C83VZA 134130016 IC50 = 15400 nM T14731 C5PFE9 134130024 IC50 = 14600 nM T14731 C3FX4R 134130170 IC50 = 57700 nM T14731 CU8FL0 134130198 IC50 = 187300 nM T14731 CJZ4F1 134130229 IC50 = 30000 nM T14731 C73SNQ 134130262 IC50 = 116000 nM T14731 CDJ7U6 134130313 IC50 = 45800 nM T14731 CJ7K0O 134130403 IC50 > 200000 nM T14731 CA3L0T 134130520 IC50 = 12400 nM T14731 C6J9NR 134130705 IC50 = 14600 nM T14731 C4R0LJ 134130733 IC50 = 5300 nM T14731 CS8X2E 134130756 IC50 = 18000 nM T14731 CQ0K3W 134130793 IC50 = 149500 nM T14731 CWV34S 134130814 IC50 = 220 nM T14731 C3M0AD 134130906 IC50 = 171000 nM T14731 C53GIN 134131007 IC50 = 39300 nM T14731 CA4CT5 134131074 IC50 = 27000 nM T14731 CP2RV4 134131255 IC50 = 133100 nM T14731 C4JHA7 134131282 IC50 = 77500 nM T14731 CM3B1R 134131317 IC50 > 900000 nM T14731 C8WD3G 134132512 IC50 = 3840 nM T14731 C2RX4P 134132760 IC50 = 1210 nM T14731 CI1UZ4 134133370 IC50 = 1080 nM T14731 C6C1OW 134137237 IC50 = 30000 nM T14731 CD0FX8 134139976 IC50 = 5900 nM T14731 C7P4OF 134141051 IC50 = 710 nM T14731 CYAK84 134141382 IC50 = 500 nM T14731 C7B5KW 134142322 IC50 = 270 nM T14731 CC4Z9Q 134143263 IC50 = 1100 nM T14731 CC59HY 134144404 IC50 = 93 nM T14731 CPKD12 134145576 IC50 = 570 nM T14731 CN15TH 134148556 IC50 = 820 nM T14731 CDBF51 134148882 IC50 = 22000 nM T14731 C53ATF 134148970 IC50 = 1270 nM T14731 CRON29 134150759 IC50 = 680 nM T14731 C8MGQ9 134153152 IC50 = 180 nM T14731 CZ8KH9 134155806 IC50 = 450 nM T14731 CO2I4C 134433618 IC50 > 300000 nM T14731 C9YPF1 134820907 IC50 > 100000 nM T14731 CZR65A 135397670 IC50 > 100000 nM T14731 C64DLE 135397680 IC50 = 100000 nM T14731 C51NFI 135420639 IC50 = 5900 nM T14731 C8F5SE 135425069 IC50 = 13000 nM T14731 CB53GJ 135443018 IC50 = 5900 nM T14731 C4KDT9 135457159 IC50 = 42400 nM T14731 CW50RD 135469837 IC50 = 89300 nM T14731 C2EF5P 135536415 EC50 = 10400 nM T14731 CG3UM8 135579320 EC50 = 7000 nM T14731 CU3G1F 135641258 EC50 = 4500 nM T14731 CE3VW5 135659046 IC50 = 37500 nM T14731 CC1L0B 135800241 IC50 = 40300 nM T14731 CT7ZX6 135800242 IC50 = 40300 nM T14731 CND1B8 135862920 IC50 = 40300 nM T14731 C98WZT 135862921 IC50 = 40300 nM T14731 CL8FY6 135867735 EC50 = 1600 nM T14731 C9LBZ5 135867742 EC50 = 1700 nM T14731 C42VRW 135867743 EC50 = 5400 nM T14731 CL92IA 135867746 EC50 = 2700 nM T14731 CWE43H 136226206 EC50 = 2000 nM T14731 CP38AV 136226207 EC50 = 55200 nM T14731 CF9R3E 136226208 EC50 = 2300 nM T14731 C12LYB 136226209 EC50 = 3400 nM T14731 CO5PQ9 136236339 IC50 = 40300 nM T14731 CAN4M5 136236340 IC50 = 40900 nM T14731 CJB12C 136236341 IC50 = 40300 nM T14731 CCJE20 136236342 IC50 = 40300 nM T14731 C1R9OX 136236343 IC50 = 40300 nM T14731 C5GIF3 136236344 IC50 = 40300 nM T14731 CIX5U1 136236345 IC50 = 40300 nM T14731 CZQI18 136236346 IC50 = 40300 nM T14731 CG7K6R 136240899 EC50 = 2600 nM T14731 CUHJ90 136240940 EC50 = 2100 nM T14731 CK5XC6 136240941 EC50 = 1800 nM T14731 CWXJ76 136240942 EC50 = 3700 nM T14731 CY0K4T 136240974 EC50 = 28100 nM T14731 CRKA87 136240975 EC50 = 2300 nM T14731 CESH75 136240976 EC50 = 900 nM T14731 CNG4Z7 136240977 EC50 = 18300 nM T14731 C0V7WJ 136241907 EC50 = 900 nM T14731 CN5S6P 136241915 EC50 = 18100 nM T14731 C7Z1GW 136241916 EC50 = 1600 nM T14731 C0XCH7 136241917 EC50 = 9600 nM T14731 C4K6OX 136241918 EC50 = 20500 nM T14731 C2ZPN0 136241927 EC50 = 8700 nM T14731 CA93FC 136241928 EC50 = 4400 nM T14731 CQ9W1P 137634939 IC50 = 54800 nM T14731 C8YK2Z 137642096 IC50 = 129000 nM T14731 C4U5WK 137644691 IC50 = 108700 nM T14731 C9FN7L 137649628 IC50 = 13830 nM T14731 CIT7K5 137658301 IC50 = 109900 nM T14731 CLW0B7 137661474 IC50 = 42120 nM T14731 CAQ62X 137701235 Ki > 10000 nM T14731 C62HXG 138319670 IC50 > 100000 nM T14731 CN2UH1 139303146 IC50 > 20000 nM T14731 CW7HG8 145960911 IC50 > 200000 nM T14731 CC0VT3 145962411 IC50 > 200000 nM T14731 CCXR94 145963449 IC50 = 5300 nM T14731 C5QIN6 145963700 IC50 > 300000 nM T14731 CX3MQ7 145965297 IC50 = 35070 nM T14731 C9XT0U 145966202 IC50 > 50000 nM T14731 C6W3YP 145966373 IC50 = 29800 nM T14731 CHQ8Z0 145967555 IC50 > 50000 nM T14731 C7ML9P 145967841 IC50 > 100000 nM T14731 CC3G2E 145970505 IC50 > 50000 nM T14731 C9CJ3Y 145971573 IC50 = 36970 nM T14731 CP1I5W 145972149 IC50 > 50000 nM T14731 CB51IT 145973739 IC50 = 97400 nM T14731 CLT69F 145975278 IC50 = 19960 nM T14731 CWD0A9 145983712 Ki > 10000 nM T14731 C56MWZ 145986208 Ki > 10000 nM T14731 C8AS1P 155512143 IC50 = 34000 nM T14731 C80DBU 155512388 IC50 > 200000 nM T14731 CPZ01A 155512728 IC50 = 11000 nM T14731 CPQ48B 155513088 IC50 = 4300 nM T14731 CM6VN5 155513154 IC50 = 26 nM T14731 CZE29G 155514745 IC50 = 1800 nM T14731 C7VC1F 155517856 IC50 > 2000 nM T14731 CU0M1P 155518467 IC50 = 50 nM T14731 CDY5H6 155519645 IC50 > 10000 nM T14731 CN78HI 155519887 IC50 = 48 nM T14731 C2M5UT 155520367 IC50 > 2000 nM T14731 C09RAW 155520570 IC50 = 1700 nM T14731 CH78ST 155523405 IC50 > 100000 nM T14731 CFH1D8 155524740 IC50 = 1000 nM T14731 C4HV9G 155525499 IC50 = 98 nM T14731 C7H6XU 155528914 IC50 = 140 nM T14731 CTH59X 155529937 IC50 > 200000 nM T14731 CX8SC4 155530876 IC50 > 2000 nM T14731 C1JKR4 155531258 IC50 = 77400 nM T14731 C9WNP0 155531613 IC50 = 1000 nM T14731 CLD19W 155539311 IC50 > 10000 nM T14731 C61BTI 155545173 IC50 = 84 nM T14731 CH30TZ 155546485 IC50 > 100000 nM T14731 C3WAN0 155550829 IC50 = 1.81 ug.mL-1 T14731 C2FZ1M 155550843 IC50 > 100000 nM T14731 C3D7GP 155554414 IC50 = 22000 nM T14731 C6FV9S 155554968 IC50 = 30000 nM T14731 CG7PH3 155555586 IC50 = 1400 nM T14731 CLA4P7 155561544 IC50 = 98 nM T14731 C7IWD4 155564228 IC50 = 450 nM T14731 C4CIL9 155564382 IC50 > 2000 nM T14731 D00LYI 135461039 IC50 = 59000 nM T14731 D02AYX 1403654 IC50 = 5300 nM T14731 D02EWM 1376646 IC50 = 55000 nM T14731 D03APP 4386 IC50 = 68000 nM T14731 D07WDQ 66541 IC50 = 870 nM T14731 D09AFM 88489 IC50 = 32000 nM T14731 D09SUO 5269 IC50 = 96200 nM T14731 D09VTJ 441298 IC50 = 15000 nM T14731 D0D5ZL 369401 IC50 = 8000 nM T14731 D0E1QP 4262314 IC50 = 1470 nM T14731 D0E3NT 2130404 IC50 = 30000 nM T14731 D0F1KR 1376645 IC50 = 67000 nM T14731 D0M5FF 5083 IC50 = 3500 nM T14731 D0TO6S 2396 IC50 = 23000 nM T14731 D0UO1E 135491748 IC50 = 13000 nM T02752 D09RGW 11753159 Ki = 6.31 nM T02752 D0W0LS 183789 IC50 > 10000 nM T02752 CPS2A1 77033 IC50 = 383 nM T02752 C7X0IR 209394 IC50 = 190 nM T02752 CQ3KO7 483339 IC50 > 1000 nM T02752 C7AP9W 483340 IC50 > 1000 nM T02752 CAB79M 483341 IC50 > 1000 nM T02752 C7XW2D 483342 IC50 > 1000 nM T02752 C7PMT6 483343 IC50 > 1000 nM T02752 CP25RI 483344 IC50 > 1000 nM T02752 CUM8T0 2729098 IC50 = 1300 nM T02752 CMT8K7 5481702 IC50 = 10000 nM T02752 CHCY06 6918496 IC50 = 0.58 nM T02752 C18KRM 6918497 IC50 = 0.58 nM T02752 CC2K1A 6995527 IC50 = 9000 nM T02752 C89QWY 6999830 IC50 > 50000 nM T02752 CG28LQ 7039308 IC50 > 20000 nM T02752 COY73G 7072714 IC50 = 6250 nM T02752 C34YGS 9797962 Ki = 90 nM T02752 CUY72A 9800669 IC50 = 8 nM T02752 C2SD3N 9804542 IC50 = 4 nM T02752 CHTN02 9818195 IC50 = 5950 nM T02752 C4KGP2 9825034 IC50 = 10 nM T02752 CVY67K 9826988 IC50 = 600 nM T02752 CVGW51 9840971 IC50 = 49 nM T02752 CYZ47C 9842640 IC50 = 200 nM T02752 C54ZSI 9845853 IC50 = 67 nM T02752 C8FPN7 9847583 IC50 = 4.4 nM T02752 CK3V7O 9868459 IC50 = 6 nM T02752 CM5R7B 9868532 IC50 = 12 nM T02752 CK7FJ6 9870185 Ki = 1.585 nM T02752 C5RP3D 9885355 IC50 = 80 nM T02752 C78BEF 9888454 IC50 = 330 nM T02752 CE13DO 9889700 IC50 = 9000 nM T02752 CDL61K 9892753 IC50 = 1 nM T02752 CEV5L0 9907041 IC50 = 16000 nM T02752 C3IPW5 9910169 Ki = 100 nM T02752 CF4VO1 9914506 Ki = 5.012 nM T02752 C78OBX 9927733 IC50 = 325 nM T02752 C24MLV 9935588 IC50 = 3900 nM T02752 CV6M7P 9951882 IC50 = 55 nM T02752 C5FJ9S 9951883 IC50 = 300 nM T02752 C4VSP8 9952288 IC50 = 563 nM T02752 C91RTG 9956238 IC50 > 10000 nM T02752 CKY24I 9957612 IC50 = 5 nM T02752 CFV43T 9972570 IC50 = 8400 nM T02752 CJ2HT6 9979012 IC50 = 1000 nM T02752 CP5JS6 9981262 IC50 = 36 nM T02752 C0FKS6 9982077 IC50 = 237 nM T02752 CH5C2N 10000888 IC50 = 750 nM T02752 CCB2G9 10003872 Ki = 50 nM T02752 CZW1M7 10005242 Ki = 12.59 nM T02752 CTDC61 10029075 IC50 = 40 nM T02752 CK63CE 10050884 IC50 = 0.3 nM T02752 C94DWF 10096657 IC50 = 1.3 nM T02752 CPH1C7 10140602 IC50 = 0.2 nM T02752 C4SHX2 10142792 IC50 = 750 nM T02752 C7YM5L 10143016 Ki = 158.49 nM T02752 CLW3J6 10151756 Ki = 39.81 nM T02752 CY4OA2 10164316 IC50 > 10000 nM T02752 CBTG57 10182382 IC50 > 10000 nM T02752 C5Z8RT 10187492 IC50 > 10000 nM T02752 CNG8I1 10194663 IC50 = 190 nM T02752 C9AJ4D 10255492 IC50 = 3 nM T02752 CW7MP5 10257335 IC50 = 535 nM T02752 CZNP37 10300214 Ki = 100 nM T02752 C7F9SZ 10322255 IC50 = 1.6 nM T02752 CWFB30 10323427 IC50 > 1000 nM T02752 CSW05N 10457573 IC50 = 2.6 nM T02752 CW2P3H 10458117 IC50 = 85 nM T02752 CVAD83 10458976 IC50 = 0.013 nM T02752 CW6K9H 10459751 IC50 = 0.7 nM T02752 CA5YI3 10474776 IC50 = 5 nM T02752 C05PCB 10591473 IC50 = 7100 nM T02752 C53DCW 10623381 IC50 = 12000 nM T02752 CMQP67 10863252 IC50 = 24 nM T02752 COAC81 10863284 IC50 = 35 nM T02752 COM0W2 10864223 IC50 = 42 nM T02752 C9EZ4N 10873705 IC50 = 79 nM T02752 CET2D1 10874167 IC50 = 1750 nM T02752 CDF2L4 10874195 IC50 = 360 nM T02752 CWK8N7 10874762 IC50 = 7 nM T02752 C61SVO 10874991 IC50 = 3900 nM T02752 C47TRP 10875472 IC50 = 3500 nM T02752 C9LO8N 10895831 IC50 = 11 nM T02752 CJWQ05 10906911 IC50 = 47 nM T02752 C6HE2M 10916572 IC50 = 4600 nM T02752 CF07JD 10917990 IC50 = 141 nM T02752 C0EM4G 10928173 IC50 = 280 nM T02752 CX1GK6 10928228 IC50 = 1750 nM T02752 CL0EY6 10928826 IC50 = 55 nM T02752 CNZ07K 10929194 IC50 = 67 nM T02752 C86DMO 10934382 IC50 = 8300 nM T02752 CCQ92I 10939210 IC50 = 3800 nM T02752 CFX5E8 10939698 IC50 = 9 nM T02752 CXT0E9 10950225 IC50 = 2800 nM T02752 CH1MV6 10962347 IC50 = 8 nM T02752 C1ZK6C 10972522 IC50 = 14 nM T02752 CX2K8E 10974378 IC50 = 1620 nM T02752 C5CI0F 10979426 IC50 = 50000 nM T02752 C2CQW9 10983106 IC50 = 2400 nM T02752 C5ZSX2 10983308 IC50 = 114 nM T02752 CP20ZE 10983419 IC50 = 17 nM T02752 CQ24OW 10983980 IC50 = 64 nM T02752 CAN36G 10983981 IC50 = 11 nM T02752 CB2CG7 10984360 IC50 = 48 nM T02752 CN87LP 10985078 IC50 = 5200 nM T02752 CZM5K3 10993686 IC50 = 750 nM T02752 CWS9J7 10995218 IC50 = 2350 nM T02752 CDO30J 10995329 IC50 = 5950 nM T02752 C48JFQ 11001953 IC50 = 2600 nM T02752 CPC19I 11004663 IC50 = 140 nM T02752 CVL3G5 11004681 IC50 = 620 nM T02752 C3GF2J 11004826 IC50 = 53 nM T02752 C6IST9 11005432 IC50 = 777 nM T02752 C20UVD 11006581 IC50 = 11 nM T02752 CGY15F 11015975 IC50 = 81 nM T02752 CS47JM 11017617 IC50 = 2 nM T02752 CK70OY 11026367 IC50 = 600 nM T02752 C82RPC 11026461 IC50 = 7600 nM T02752 CJGS81 11026634 IC50 = 180 nM T02752 C9ETA8 11037869 IC50 = 125 nM T02752 CNE74S 11037958 IC50 = 32 nM T02752 C4APJ9 11038430 IC50 = 2 nM T02752 CZ3CB6 11048445 IC50 = 450 nM T02752 C4E7CJ 11048458 IC50 = 277 nM T02752 C9UK2E 11049424 IC50 = 8300 nM T02752 CIA6O3 11059280 IC50 = 310 nM T02752 C8DY3J 11059385 IC50 = 153 nM T02752 CD2E4K 11059789 IC50 = 11 nM T02752 CVX0M9 11060510 IC50 = 6100 nM T02752 C8JG0H 11060814 IC50 = 9800 nM T02752 CL82DR 11069916 IC50 = 750 nM T02752 COC29P 11070954 IC50 = 8 nM T02752 CH0DL9 11072063 IC50 = 7600 nM T02752 CSUH61 11072275 IC50 = 5300 nM T02752 C89VIY 11081509 IC50 = 529 nM T02752 CFG06R 11082578 IC50 = 5700 nM T02752 CCD3L5 11091447 IC50 = 450 nM T02752 CV6E7Q 11101888 IC50 = 11000 nM T02752 C43FIU 11102400 IC50 = 4650 nM T02752 CCN74A 11103844 IC50 = 21 nM T02752 C90YHK 11104005 IC50 = 2200 nM T02752 CBU6C5 11112528 IC50 = 361 nM T02752 C4FB5K 11113940 IC50 = 20 nM T02752 CZ9U7O 11124782 IC50 = 2400 nM T02752 C9P3ME 11133428 IC50 = 3400 nM T02752 CIP20Q 11134412 IC50 = 410 nM T02752 CDKJ18 11134936 IC50 = 2 nM T02752 CZH8W1 11144348 IC50 = 450 nM T02752 CKZR60 11145481 IC50 = 3700 nM T02752 C0VCM7 11154845 IC50 = 1.6 nM T02752 C49DJB 11156406 IC50 = 0.9 nM T02752 CTN28W 11167549 IC50 = 1.2 nM T02752 CFG0U2 11169258 IC50 = 0.042 nM T02752 CJ4P0Q 11179351 IC50 = 2.2 nM T02752 CT2J3Z 11179592 IC50 = 6 nM T02752 CK5AM4 11179794 Ki = 20 nM T02752 C4GAT3 11213416 IC50 = 1 nM T02752 C42SVZ 11213457 IC50 = 3.7 nM T02752 C30WRJ 11214422 Ki = 18 nM T02752 CB0HV1 11214474 IC50 = 4 nM T02752 C2PR4C 11224689 IC50 = 9 nM T02752 C8T7PC 11226588 IC50 = 60 nM T02752 CA39QR 11227406 IC50 = 0.034 nM T02752 C58JIR 11236236 IC50 = 9 nM T02752 C07EZW 11236950 IC50 = 0.6 nM T02752 C2LNX0 11247999 IC50 = 14 nM T02752 C3P2DG 11259591 IC50 = 4.6 nM T02752 CQ6KW0 11272103 IC50 = 0.01 nM T02752 CIR02K 11282712 IC50 = 41 nM T02752 C8EF0Y 11283679 Ki = 15 nM T02752 C06TUD 11285791 IC50 = 2400 nM T02752 C4JNV9 11306550 IC50 = 1.3 nM T02752 CBP52U 11316656 IC50 = 5 nM T02752 CLN4K5 11328714 IC50 = 2 nM T02752 C1A5ET 11329244 IC50 = 0.03 nM T02752 CM3O5G 11340670 IC50 = 0.015 nM T02752 C5F8DG 11351206 IC50 = 1.8 nM T02752 CD98SB 11360133 Ki = 28 nM T02752 CF2E4B 11363005 IC50 = 1.4 nM T02752 CLI6Y2 11363006 IC50 = 1 nM T02752 C75ROL 11373714 IC50 = 1.9 nM T02752 C0O8VA 11385178 IC50 = 10 nM T02752 CPO48X 11385474 IC50 = 78 nM T02752 CN0SU2 11385766 IC50 = 0.364 nM T02752 CZ9RO8 11386642 Ki = 23 nM T02752 CO6E3D 11396851 IC50 = 14 nM T02752 C7I6UM 11396966 IC50 = 31 nM T02752 CC02JA 11396995 IC50 = 12 nM T02752 C4I3RD 11397114 IC50 = 0.06 nM T02752 C04CJR 11397231 Ki = 9 nM T02752 CP21VU 11398022 IC50 = 0.25 nM T02752 CQ7ZP0 11408397 IC50 = 29 nM T02752 C7E6IT 11409583 IC50 = 1.1 nM T02752 C4M1LX 11419003 IC50 = 1.9 nM T02752 CQY2D8 11430170 IC50 = 2.5 nM T02752 CUW4P9 11442162 IC50 = 1.4 nM T02752 CPIU38 11442439 IC50 = 4 nM T02752 CG58SO 11444350 Ki = 19.95 nM T02752 CEA2J7 11454015 IC50 = 1.6 nM T02752 CQ1RF9 11454941 IC50 = 0.1 nM T02752 CK4S8F 11465468 IC50 = 3 nM T02752 CAG67M 11466397 Ki = 3.3 nM T02752 CV3KP0 11477384 IC50 = 1.8 nM T02752 CF6QA7 11477767 Ki = 7.7 nM T02752 C89GBJ 11487192 IC50 = 2.7 nM T02752 C1QGD0 11488078 IC50 = 0.045 nM T02752 CETO93 11511522 IC50 = 65 nM T02752 C0SVJ7 11540776 Ki = 30 nM T02752 CP5OU4 11609863 IC50 = 14500 nM T02752 CJ5ZS3 11698698 IC50 = 0.6 nM T02752 C3KU0D 11722772 IC50 = 3800 nM T02752 CB34MH 11729258 IC50 = 14100 nM T02752 C24ZXA 11730610 IC50 = 228 nM T02752 C7QER1 11730796 IC50 = 1 nM T02752 C9D2CH 11732727 IC50 = 249 nM T02752 CVB47P 11733139 IC50 = 49 nM T02752 C58TMP 11733617 IC50 = 3 nM T02752 CVLM30 11734303 IC50 = 3000 nM T02752 CPG15O 11743399 IC50 > 10000 nM T02752 CK16GS 11750808 IC50 = 2.3 nM T02752 CG39UJ 11751629 IC50 = 1.7 nM T02752 CYX08E 11762084 IC50 = 9200 nM T02752 CF3L4U 11762511 IC50 = 2 nM T02752 CK76RF 11762865 IC50 = 2650 nM T02752 CL9P2V 11763035 IC50 = 8 nM T02752 CSX85G 11811443 IC50 = 900 nM T02752 CLME86 11812728 IC50 = 7350 nM T02752 C4E1CI 11812807 IC50 = 21 nM T02752 COZ69K 11813735 IC50 = 2230 nM T02752 CT8D3H 11814253 IC50 = 19300 nM T02752 CO23LC 11825113 IC50 = 2600 nM T02752 CLX43D 11826382 IC50 = 1300 nM T02752 C96ZJD 11828013 IC50 = 8300 nM T02752 C6QN3V 11828215 IC50 = 2200 nM T02752 CX6Y7W 11952524 Ki = 67 nM T02752 CA97XF 11952525 Ki = 120 nM T02752 C49USB 11952526 Ki = 4.9 nM T02752 CK13QD 11953409 IC50 = 0.068 nM T02752 CQFM31 11966687 IC50 = 1 nM T02752 CAW2Y1 12000105 IC50 = 2 nM T02752 CNO57E 12001832 Ki = 0.5012 nM T02752 CX27OB 15907328 IC50 = 18700 nM T02752 CH8K6G 16040671 Ki = 0.631 nM T02752 C9UYE0 16126667 IC50 = 1.7 nM T02752 CY0UI3 16681693 Ki = 1.8 nM T02752 CK3WA5 16747712 IC50 = 1.3 nM T02752 C8QFZ1 17963141 Ki = 125.89 nM T02752 CP72GT 17963153 Ki = 25.12 nM T02752 C67NRA 17963183 Ki = 6.31 nM T02752 CHW4F9 17963196 Ki = 39.81 nM T02752 C8MJG3 17963199 Ki = 630.96 nM T02752 C1H3UD 17963201 Ki = 0.631 nM T02752 CJS35W 17963208 Ki = 31.62 nM T02752 CBNK23 17963226 Ki = 7.943 nM T02752 C5ZT8C 17963227 Ki = 100 nM T02752 C9EVG1 17963258 Ki = 50.12 nM T02752 CQ7WR1 17963315 Ki = 15.85 nM T02752 C2V6WP 17963332 Ki = 25.12 nM T02752 COCE85 17963334 Ki = 19.95 nM T02752 C8KRN7 17963336 Ki = 100 nM T02752 CRYU86 17963347 Ki = 31.62 nM T02752 C2PWS7 17963363 Ki = 7.943 nM T02752 CWY0T6 17989653 Ki = 100 nM T02752 CZK1E8 20576924 IC50 = 1100 nM T02752 CX7FG2 20613253 IC50 = 1700 nM T02752 C81FRQ 20636465 IC50 = 4.3 nM T02752 CK7HS6 21362416 IC50 = 2.2 nM T02752 C8OHV9 21362425 IC50 = 2 nM T02752 CV39JS 22022826 IC50 = 1800 nM T02752 C3TSH9 22022834 IC50 = 5300 nM T02752 C53NIP 22143196 IC50 = 19.7 nM T02752 C1Q4LP 22257689 IC50 = 500 nM T02752 CX7F9I 22393282 IC50 = 10 nM T02752 CVE4C2 22393287 IC50 = 5 nM T02752 CUW8L9 22393307 IC50 = 200 nM T02752 CE80BF 22393315 IC50 = 41 nM T02752 CK37OM 22393329 IC50 = 29 nM T02752 C0SF1T 22393333 IC50 = 400 nM T02752 CQ8J9F 22393339 IC50 = 20 nM T02752 CID72N 22393362 IC50 = 200 nM T02752 C79NHX 22393366 IC50 = 200 nM T02752 C2P0MY 22393370 IC50 = 500 nM T02752 CSH1Y2 22393378 IC50 = 300 nM T02752 C1BL8Z 22393395 IC50 = 38 nM T02752 C3DX2Z 22393396 IC50 = 243 nM T02752 CH02UC 22393398 IC50 = 500 nM T02752 CX64QZ 22393419 IC50 = 30 nM T02752 CYB14S 22393428 IC50 = 400 nM T02752 C3RZ5G 22393430 IC50 = 20 nM T02752 C5WRI7 22393436 IC50 = 100 nM T02752 CQ0JS3 22393469 IC50 = 20 nM T02752 CD80BP 22393474 IC50 = 70 nM T02752 CL5D9B 22397436 Ki = 50.12 nM T02752 CDJ12S 22397445 Ki = 10 nM T02752 CPH6L4 22966050 IC50 = 7 nM T02752 C7L0UG 22966052 IC50 = 386 nM T02752 CD14YL 23102733 Ki = 79.43 nM T02752 CU1T8V 23102749 Ki = 12.59 nM T02752 CDW58L 23497297 IC50 = 260 nM T02752 C65QTZ 23509664 IC50 = 1600 nM T02752 CC5QG6 23509693 IC50 = 40 nM T02752 CA9LH1 23509695 IC50 = 50 nM T02752 C4LGP9 23509697 IC50 = 30 nM T02752 CC60DR 23657036 IC50 = 12 nM T02752 C25HKJ 24758044 IC50 > 30000 nM T02752 CX79IO 24882359 IC50 = 20 nM T02752 COJ6M7 24937092 Ki = 82 nM T02752 CFX5V9 24937215 Ki = 61 nM T02752 CI8B1E 25024650 Ki = 5 nM T02752 C2S0FP 25024651 Ki = 16 nM T02752 C7GME3 25024849 Ki = 54 nM T02752 CKN6Y0 25024850 Ki = 60 nM T02752 CAH8P4 25032958 IC50 = 0.5 nM T02752 CKIR47 25056323 Ki = 62 nM T02752 CRMF16 25056324 Ki = 80 nM T02752 COSJ47 25056325 Ki = 316 nM T02752 C54LQF 25230828 IC50 > 50000 nM T02752 C2A7ZX 25751147 EC50 = 1500 nM T02752 C4M1KP 38347547 EC50 = 1400 nM T02752 C0J4FI 43957010 Ki = 7750 nM T02752 C4J6IN 44273640 IC50 = 1000 nM T02752 C7MRP6 44281349 IC50 > 25000 nM T02752 C45QUS 44281365 IC50 > 25000 nM T02752 CUQ95A 44281373 IC50 > 25000 nM T02752 CT5IO4 44281489 IC50 > 33000 nM T02752 CF0CJ2 44281521 IC50 = 3 nM T02752 CX2KF1 44281522 IC50 = 33000 nM T02752 CL4Q6F 44281523 IC50 = 4000 nM T02752 C4N5MW 44281525 IC50 = 1700 nM T02752 CUT37W 44281598 IC50 > 33000 nM T02752 CJE5T3 44281612 IC50 = 190 nM T02752 CYLO98 44281667 IC50 = 300 nM T02752 C6M1AT 44281668 IC50 = 27 nM T02752 CNDM47 44281673 IC50 = 116 nM T02752 CW72RQ 44281686 IC50 = 666 nM T02752 CB48QR 44281706 IC50 = 400 nM T02752 CH3I6F 44281754 IC50 = 800 nM T02752 CLB43T 44281755 IC50 = 500 nM T02752 C5AH1J 44281774 IC50 = 700 nM T02752 CR40YV 44281775 IC50 = 65 nM T02752 CEF45P 44281789 IC50 = 18 nM T02752 C27ODI 44281790 IC50 = 57 nM T02752 CIM1A2 44281791 IC50 = 21 nM T02752 CD5H9W 44281793 IC50 = 17000 nM T02752 CFY2G1 44281794 IC50 = 600 nM T02752 CQNZ37 44281852 IC50 = 45 nM T02752 CC2T7Y 44281859 IC50 = 3 nM T02752 C5JWR1 44281872 IC50 = 7700 nM T02752 C89IHR 44281891 IC50 = 18000 nM T02752 CVZ1N5 44281915 IC50 > 1220 nM T02752 C1WZG9 44281916 IC50 > 33000 nM T02752 CV63NE 44281943 IC50 = 22500 nM T02752 CEL15O 44281944 IC50 = 45 nM T02752 C9OK7H 44281951 IC50 = 663 nM T02752 CTB3F0 44281966 IC50 = 32000 nM T02752 C2G0YU 44281975 IC50 = 20 nM T02752 CH3J9N 44281987 IC50 = 600 nM T02752 CU51QR 44281999 IC50 = 500 nM T02752 C7HZ0M 44282005 IC50 = 250 nM T02752 C5S2NQ 44282006 IC50 = 15 nM T02752 CSOY75 44282030 IC50 = 213 nM T02752 CR39VI 44282031 IC50 = 1125 nM T02752 C73SAY 44282047 IC50 = 90 nM T02752 CKFI08 44282048 IC50 = 125 nM T02752 C75JZM 44282280 IC50 = 383 nM T02752 CHF42Q 44282379 IC50 > 33000 nM T02752 C6FT0O 44282385 IC50 = 12500 nM T02752 C13YSW 44289699 IC50 = 49 nM T02752 CDO12U 44289701 IC50 = 0.7 nM T02752 C8QW3Z 44289713 IC50 = 2.4 nM T02752 CB9L7J 44289715 IC50 = 1 nM T02752 CQO8L7 44289741 IC50 = 1.2 nM T02752 C8EY2C 44289762 IC50 = 31 nM T02752 COS7M9 44289763 IC50 = 19 nM T02752 CB8CA1 44289877 IC50 = 3.6 nM T02752 C7FHP0 44289910 IC50 = 3.1 nM T02752 C6UR1Q 44289919 IC50 = 2.6 nM T02752 CMUT04 44289926 IC50 = 1.2 nM T02752 CQ4Y0G 44289927 IC50 = 0.6 nM T02752 CJ1KV7 44289959 IC50 = 39 nM T02752 CUZ7W4 44290018 IC50 = 1.2 nM T02752 CIYO50 44290019 IC50 = 3.1 nM T02752 C8JL4Z 44290020 IC50 = 7.1 nM T02752 C1TF0N 44290029 IC50 = 7.9 nM T02752 CHM25N 44290039 IC50 = 2.5 nM T02752 C15ZHK 44290040 IC50 = 39 nM T02752 CVQS56 44290041 IC50 = 56 nM T02752 CB2QI4 44290100 IC50 = 0.9 nM T02752 C9TQY8 44295065 IC50 = 6800 nM T02752 CS4IV9 44295102 IC50 = 5100 nM T02752 C4LM0C 44295118 IC50 = 8100 nM T02752 CA69UI 44295130 IC50 = 500 nM T02752 CSI6J1 44295145 IC50 = 1500 nM T02752 C8R5TX 44295201 IC50 = 60 nM T02752 C29TPL 44295230 IC50 = 5500 nM T02752 C1JGI8 44295259 IC50 = 3900 nM T02752 CF53GA 44295264 IC50 = 100 nM T02752 CTO78G 44295267 IC50 = 200 nM T02752 CF67CX 44295282 IC50 = 7 nM T02752 CK39HF 44295286 IC50 = 50 nM T02752 CG6OA1 44295288 IC50 = 70 nM T02752 C2Q8XF 44295304 IC50 = 200 nM T02752 C0E2QB 44295306 IC50 = 20 nM T02752 CV6Z9T 44295326 IC50 = 9 nM T02752 C7DXZ2 44295327 IC50 = 89 nM T02752 CAE81F 44295328 IC50 = 60 nM T02752 CZ86IO 44295352 IC50 = 1200 nM T02752 CM5F0L 44295353 IC50 = 800 nM T02752 CUO2N1 44295354 IC50 = 1600 nM T02752 CU7R1B 44295362 IC50 = 30 nM T02752 C68LDM 44295364 IC50 = 50 nM T02752 CM9C8A 44295372 IC50 = 1200 nM T02752 CJ79ZM 44295374 IC50 = 1200 nM T02752 CIXU43 44295375 IC50 = 4800 nM T02752 CXN92L 44295405 IC50 = 100 nM T02752 CB05IM 44295406 IC50 = 200 nM T02752 CJ6XP3 44295407 IC50 = 6600 nM T02752 C4I8BO 44295408 IC50 = 11000 nM T02752 CVRP83 44295409 IC50 = 25600 nM T02752 CF19LT 44295433 IC50 = 260 nM T02752 CZXG95 44295434 IC50 = 30 nM T02752 C0C2TL 44295435 IC50 = 10100 nM T02752 C04HZL 44295462 IC50 = 1 nM T02752 CXD5M0 44295463 IC50 = 6400 nM T02752 CRKA28 44295470 IC50 = 530 nM T02752 CPVT86 44295479 IC50 = 240 nM T02752 CFH7O5 44295480 IC50 = 170 nM T02752 CTB58O 44295485 IC50 = 5 nM T02752 C4N3RA 44295486 IC50 = 1100 nM T02752 CV5YL8 44295487 IC50 = 3700 nM T02752 C29RIS 44295499 IC50 = 250 nM T02752 CU3G7O 44295510 IC50 = 700 nM T02752 C7A0SB 44295528 IC50 = 500 nM T02752 C0EQ8H 44295529 IC50 = 1000 nM T02752 CJ92CM 44295536 IC50 = 80 nM T02752 CF5G8T 44295543 IC50 = 90 nM T02752 CZH6B0 44295544 IC50 = 1300 nM T02752 CZ09EM 44295554 IC50 = 40 nM T02752 CR4OZ0 44295555 IC50 = 20 nM T02752 CXNQ07 44295558 IC50 = 8300 nM T02752 CMZP50 44295566 IC50 = 20 nM T02752 CUJ90M 44295567 IC50 = 100 nM T02752 CG6PA4 44295591 IC50 = 7 nM T02752 CB6DZ9 44295622 IC50 = 50 nM T02752 CD51RU 44295641 IC50 = 50 nM T02752 CC0OQ6 44295648 IC50 = 20 nM T02752 CEBF67 44295664 IC50 = 100 nM T02752 C8G5SI 44295672 IC50 = 50 nM T02752 C49EYA 44295674 IC50 = 200 nM T02752 CX2J3A 44295686 IC50 = 2300 nM T02752 CZD7Y5 44346022 IC50 > 200000 nM T02752 CUOL80 44346023 IC50 = 7800 nM T02752 CT7ZD5 44346153 IC50 = 4.4 nM T02752 CJH18V 44346154 IC50 = 12 nM T02752 C52WRD 44346178 IC50 = 8500 nM T02752 C6L8EA 44346194 IC50 = 11 nM T02752 C71AVR 44346210 IC50 = 2.4 nM T02752 C5U9LB 44346211 IC50 = 500 nM T02752 C9YLD5 44346218 IC50 > 200000 nM T02752 C0S3TJ 44349204 IC50 = 12000 nM T02752 CC43UM 44349614 IC50 = 2000 nM T02752 CI0T4N 44349617 IC50 = 1000 nM T02752 C5X8LV 44386406 IC50 = 350 nM T02752 CAG49K 44387837 IC50 = 12 nM T02752 C8ZOD7 44387842 IC50 = 2.6 nM T02752 CV13WL 44387847 Ki = 830 nM T02752 C30EYG 44387850 IC50 = 9 nM T02752 C9T3JK 44387853 Ki = 832 nM T02752 CSXI26 44387856 IC50 = 3 nM T02752 CX5DN3 44387857 Ki = 932 nM T02752 C7V4GE 44389669 Ki = 103 nM T02752 C7YJK4 44389674 Ki = 119 nM T02752 COJG58 44389675 Ki = 41 nM T02752 CRGW08 44389677 Ki = 68 nM T02752 C84MUS 44389678 Ki = 1002 nM T02752 CUZ90F 44389683 Ki = 56 nM T02752 C4MJZ0 44389684 Ki = 66 nM T02752 C9T6VC 44389685 Ki = 100 nM T02752 CX4Z7R 44389688 Ki = 14 nM T02752 C0SY4V 44389690 Ki = 2255 nM T02752 CFK64L 44389695 Ki = 142 nM T02752 CGJ9Z4 44389698 Ki = 251 nM T02752 CC2QO5 44389699 Ki = 122 nM T02752 CLE63T 44389704 Ki = 29 nM T02752 CNX0O6 44389709 Ki = 136 nM T02752 CLU38C 44389712 Ki = 145 nM T02752 CPN83Y 44389719 Ki = 111 nM T02752 CS6PI7 44389721 Ki = 140 nM T02752 CK6U1C 44389722 Ki = 164 nM T02752 CR3ZJ4 44389725 Ki = 46 nM T02752 C2LEP5 44389729 Ki = 938 nM T02752 C5H0LZ 44389730 Ki = 191 nM T02752 CSM8F5 44389732 Ki = 792 nM T02752 C3CZM6 44389735 Ki = 458 nM T02752 C5G1UZ 44389736 Ki = 46 nM T02752 CE0K6Y 44389737 Ki = 30 nM T02752 CHX7B2 44389738 Ki = 33 nM T02752 CU27GH 44389744 Ki = 40 nM T02752 CJAW63 44389747 Ki = 128 nM T02752 C7QP5J 44389750 Ki = 111 nM T02752 C02HRT 44389751 Ki = 504 nM T02752 CYT25L 44389752 Ki = 38 nM T02752 C7MZ9O 44389765 Ki = 48 nM T02752 CLB78G 44389770 Ki = 205 nM T02752 CO62TI 44389784 Ki = 34 nM T02752 C5PC0E 44389790 Ki = 86 nM T02752 C9GLB8 44389832 Ki = 26 nM T02752 CCX2T9 44389868 Ki = 331 nM T02752 CX7Y5U 44389910 Ki = 35 nM T02752 CIS01D 44390837 IC50 = 1.9 nM T02752 CUE9X4 44390838 IC50 = 0.7 nM T02752 CNV34Z 44390842 IC50 = 5 nM T02752 CBAY82 44390843 IC50 = 120 nM T02752 CKJF03 44390848 IC50 = 12 nM T02752 CUH1C4 44390851 IC50 = 15 nM T02752 CM3S8Q 44390857 IC50 = 380 nM T02752 CHP3M2 44390858 IC50 = 54 nM T02752 CD3PO1 44390859 IC50 = 5.5 nM T02752 CI1C7V 44390867 IC50 = 14 nM T02752 CF85AM 44390882 IC50 = 9.7 nM T02752 CZN5V1 44390883 IC50 = 1.2 nM T02752 CU4X2M 44390891 IC50 = 13 nM T02752 C7LSA6 44390893 IC50 = 82 nM T02752 C8Y7CG 44390894 IC50 = 2.2 nM T02752 C80DSH 44390898 IC50 = 7.9 nM T02752 C6RH7W 44390911 IC50 = 5.5 nM T02752 CA89GO 44390919 IC50 = 3.7 nM T02752 CTSY03 44390927 IC50 = 2.2 nM T02752 CTH5M7 44390931 IC50 = 350 nM T02752 C2X8CE 44390938 IC50 = 1.8 nM T02752 CE52QO 44390945 IC50 = 1.6 nM T02752 CZ2LJ4 44390949 IC50 = 230 nM T02752 CQF9R7 44390954 IC50 = 3.2 nM T02752 COQ07N 44390955 IC50 = 0.63 nM T02752 C9H5VB 44390964 IC50 = 3.6 nM T02752 CPQ6T2 44390970 IC50 = 3 nM T02752 C47YOP 44390971 IC50 = 3 nM T02752 CL9EU8 44390978 IC50 = 6 nM T02752 CKC9B2 44391160 Ki = 1200 nM T02752 CNK1L3 44391170 Ki = 76 nM T02752 C9SL3J 44391171 Ki = 110 nM T02752 CDZ6J2 44391176 Ki = 260 nM T02752 CNP8M6 44391177 Ki = 350 nM T02752 CUC80P 44391192 Ki = 360 nM T02752 CB18AV 44391212 Ki = 3900 nM T02752 C9H7WY 44391213 Ki = 310 nM T02752 C0OAN9 44391235 Ki = 6100 nM T02752 C7V5ZS 44391236 Ki = 28 nM T02752 CN2I5F 44391240 Ki = 7900 nM T02752 C0ZL1C 44391247 Ki = 35 nM T02752 CDSW43 44391252 Ki = 290 nM T02752 C5QD2K 44391258 Ki = 1800 nM T02752 CQA2P8 44391268 Ki = 930 nM T02752 CKB3V5 44391276 Ki = 1400 nM T02752 CB9TW8 44391277 Ki = 270 nM T02752 C4GUH1 44391282 Ki = 820 nM T02752 CIG80M 44391296 Ki = 1600 nM T02752 C5MAK7 44391297 Ki = 1400 nM T02752 CV51YA 44391307 Ki = 1400 nM T02752 C5O6UQ 44391312 Ki = 4500 nM T02752 CQVS25 44391317 Ki = 2900 nM T02752 CQSL10 44391318 Ki = 1700 nM T02752 CJO61S 44391319 Ki = 720 nM T02752 C6X4ZT 44391329 Ki = 3200 nM T02752 CN7S8A 44391330 Ki = 140 nM T02752 COWH17 44391331 Ki = 250 nM T02752 CP92HS 44391800 Ki = 403 nM T02752 CNB3T2 44399272 Ki = 34 nM T02752 CMIP01 44399290 Ki = 767 nM T02752 CH4PX6 44399303 Ki = 7.3 nM T02752 C13GTL 44399331 Ki = 48 nM T02752 CN2TG8 44399332 Ki = 74.3 nM T02752 C4OFS8 44399368 Ki = 60 nM T02752 CFQ8M6 44399385 Ki = 29 nM T02752 CE17VT 44399389 Ki = 47 nM T02752 C2BC8U 44399395 Ki = 50 nM T02752 CKA8Z7 44399407 Ki = 86 nM T02752 CT2ND5 44399442 Ki = 92 nM T02752 CN7P4U 44399443 Ki = 391 nM T02752 COC1Z3 44399469 Ki = 23 nM T02752 C3JOG2 44399479 Ki = 99 nM T02752 CA39RL 44399482 Ki = 36 nM T02752 C85JDH 44399524 Ki = 58 nM T02752 CS03WY 44399537 Ki = 95 nM T02752 C9Q8MW 44399538 Ki = 180 nM T02752 CT6UD8 44399552 Ki = 533 nM T02752 C79WRF 44399567 Ki = 80 nM T02752 CNU42C 44399573 Ki = 107 nM T02752 CJC02L 44399574 Ki = 398 nM T02752 C9F3HC 44400944 Ki = 435 nM T02752 C2FMO7 44400945 Ki = 11200 nM T02752 CXG4O3 44400948 Ki = 326 nM T02752 CW0ZF3 44400949 Ki = 895 nM T02752 C0DEI5 44400950 Ki = 3810 nM T02752 CI54TN 44400953 Ki = 1070 nM T02752 CF1K4R 44400954 Ki = 2050 nM T02752 C5XNL3 44400972 Ki = 11600 nM T02752 C1UBK5 44400973 Ki = 1530 nM T02752 C6ZTW0 44400974 Ki = 8850 nM T02752 CYP34S 44400977 Ki = 429 nM T02752 CVI7H9 44400978 Ki = 972 nM T02752 C02TWQ 44400982 Ki = 216 nM T02752 C80ZLG 44400983 Ki = 9830 nM T02752 C4QB5T 44400990 Ki = 296 nM T02752 CE28PO 44400991 Ki = 768 nM T02752 CWKH19 44400992 Ki = 1250 nM T02752 CCIP06 44400995 Ki = 1720 nM T02752 C20GPY 44401004 Ki = 1200 nM T02752 CL0Z5N 44401005 Ki = 6000 nM T02752 CY0WP9 44401011 Ki = 34900 nM T02752 CJ26MT 44401012 Ki = 5380 nM T02752 CM4EW2 44401025 Ki = 605 nM T02752 C4AVR9 44401031 Ki = 349 nM T02752 CHXW09 44401032 Ki = 910 nM T02752 CIG9M6 44401037 Ki = 479 nM T02752 CD9GJ2 44401047 Ki = 179 nM T02752 C3SR0L 44401048 Ki = 545 nM T02752 CSF0J8 44401052 Ki = 1670 nM T02752 CW0F2L 44401053 Ki = 11700 nM T02752 CQ3B9K 44401055 Ki = 1030 nM T02752 CCB9O7 44401056 Ki = 1980 nM T02752 CO6US3 44401062 Ki = 1080 nM T02752 CD3QP2 44401063 Ki = 3540 nM T02752 C5VPL8 44401067 Ki = 2250 nM T02752 CQ10VA 44401069 Ki = 62500 nM T02752 CZ9J0B 44401070 Ki = 8020 nM T02752 C4R2AS 44401083 Ki = 344 nM T02752 CU5L4W 44401085 Ki = 782 nM T02752 C0T4IY 44401086 Ki = 1460 nM T02752 C5HGS8 44401088 Ki = 393 nM T02752 C3RX0K 44401089 Ki = 929 nM T02752 CY8W7X 44401094 Ki = 8970 nM T02752 CKEZ69 44401108 Ki = 10700 nM T02752 C1JGM0 44401109 Ki = 231 nM T02752 C2HMG6 44401110 Ki = 629 nM T02752 C91NCU 44401111 Ki = 1120 nM T02752 CZ3T8N 44401117 Ki = 26900 nM T02752 C07QVU 44401123 IC50 = 2 nM T02752 CBS23V 44401128 Ki = 1130 nM T02752 C2PVJ0 44401129 Ki = 4730 nM T02752 CCY18B 44401132 Ki = 5180 nM T02752 CAO13E 44401135 Ki = 129 nM T02752 CUR95G 44401136 Ki = 517 nM T02752 CAW15F 44401145 Ki = 5390 nM T02752 C80LHV 44401146 Ki = 484 nM T02752 C4HBN8 44401154 Ki = 346 nM T02752 C2SXC0 44401155 Ki = 897 nM T02752 CWBC80 44401160 Ki = 3350 nM T02752 C2PXD9 44401172 Ki = 1580 nM T02752 CE34PF 44401173 Ki = 10500 nM T02752 C9PRX5 44401175 Ki = 477 nM T02752 CLI9V6 44401176 Ki = 987 nM T02752 CV1Z3U 44401177 Ki = 312 nM T02752 CZ4C7D 44401182 Ki = 313 nM T02752 CS8TD4 44401183 Ki = 1310 nM T02752 CNE4A5 44401188 Ki = 1770 nM T02752 C9E8LT 44401189 Ki = 40200 nM T02752 CLC1V4 44401192 Ki = 10300 nM T02752 CZ3P0F 44401202 Ki = 1310 nM T02752 CPLO40 44401203 Ki = 6360 nM T02752 C80KOQ 44401206 Ki = 350 nM T02752 C3WZ1A 44401209 Ki = 5550 nM T02752 C2CP8R 44401225 Ki = 224 nM T02752 CH5P8G 44401226 Ki = 597 nM T02752 CIE0W7 44401227 Ki = 1040 nM T02752 CE4MK0 44401234 Ki = 914 nM T02752 CMV92K 44401235 Ki = 1710 nM T02752 C1JSR8 44401247 Ki = 1110 nM T02752 CQ24VI 44401248 Ki = 3650 nM T02752 CYB3D8 44401251 Ki = 14800 nM T02752 C85SCJ 44401252 Ki = 21800 nM T02752 CYKX53 44401255 Ki = 118 nM T02752 CATV38 44401256 Ki = 488 nM T02752 C35ZGL 44401328 IC50 = 1.9 nM T02752 CNJ1E3 44401561 IC50 = 23 nM T02752 CXA51W 44419295 IC50 = 0.9 nM T02752 CLA67J 44419296 IC50 = 1.3 nM T02752 C82VQX 44419298 IC50 = 0.9 nM T02752 CRAK93 44419299 IC50 = 3.6 nM T02752 CZT81O 44419300 IC50 = 2.3 nM T02752 C2WDJ5 44419301 IC50 = 1.9 nM T02752 C85OTF 44419303 IC50 = 12.4 nM T02752 CRL6M4 44419305 IC50 = 1380 nM T02752 CZ5O8Y 44419306 IC50 = 3.9 nM T02752 CXP1A6 44419308 IC50 = 5.8 nM T02752 CM3K1F 44419314 IC50 = 13 nM T02752 CYV36S 44419322 IC50 = 185 nM T02752 CY2Z7X 44419323 IC50 = 142 nM T02752 CG8F3J 44419327 IC50 = 6 nM T02752 CJR7P1 44419328 IC50 = 1.4 nM T02752 C7DQL6 44419331 IC50 = 0.5 nM T02752 CVMF25 44419335 IC50 = 2.5 nM T02752 C59ZPV 44419340 IC50 = 4.1 nM T02752 C71CPW 44419344 IC50 = 0.7 nM T02752 CM1WZ9 44419345 IC50 = 1 nM T02752 C0NY7S 44440393 IC50 = 158 nM T02752 CE24WK 44440394 IC50 = 32 nM T02752 CEA4M1 44440396 IC50 = 25 nM T02752 CD9ER1 44440398 IC50 = 100 nM T02752 C08UCK 44440402 IC50 = 20 nM T02752 CG2N8X 44440411 IC50 = 100 nM T02752 CSL2E4 44440412 IC50 = 40 nM T02752 CM5O3W 44440413 IC50 = 63 nM T02752 CCV4I0 44440414 IC50 = 100 nM T02752 CAI8C7 44440417 IC50 = 100 nM T02752 CS8TO3 44440419 IC50 = 158 nM T02752 C0UCI6 44440420 IC50 = 100 nM T02752 CI4AO7 44440421 IC50 = 79 nM T02752 CZ2LN9 44440422 IC50 = 2500 nM T02752 CGR1F7 44440423 IC50 = 400 nM T02752 C28MNA 44440424 IC50 = 100 nM T02752 CHK61S 44440426 IC50 = 100 nM T02752 C9YBH5 44440427 IC50 = 250 nM T02752 C6CYF7 44440429 IC50 = 200 nM T02752 C8MI5L 44440431 IC50 = 6.3 nM T02752 CV4Z8R 44440434 IC50 = 2500 nM T02752 CI0VR6 44440435 IC50 = 1000 nM T02752 CHI4O8 44440437 IC50 = 12 nM T02752 CT90QL 44440438 IC50 > 10000 nM T02752 C1VYA9 44440440 IC50 = 2500 nM T02752 CRCH37 44440445 IC50 = 200 nM T02752 CWCY76 44442586 IC50 > 10000 nM T02752 C89VZB 44442587 IC50 > 10000 nM T02752 C6M2TZ 44442590 IC50 = 10000 nM T02752 C93GZU 44442593 IC50 > 10000 nM T02752 CU43VX 44442598 IC50 > 10000 nM T02752 C84AZN 44442599 IC50 = 1500 nM T02752 CWE9P2 44445839 IC50 = 1.7 nM T02752 CH7W8P 44445840 IC50 = 2 nM T02752 CY2KD0 44445842 IC50 = 1 nM T02752 C5W8MO 44445843 IC50 = 6 nM T02752 C5OYU7 44445845 IC50 = 0.1 nM T02752 C81EKO 44445846 IC50 = 9.2 nM T02752 CY7XD2 44445847 IC50 = 0.075 nM T02752 CRV2Y7 44445849 IC50 = 2.6 nM T02752 CSC7N1 44445850 IC50 = 7.6 nM T02752 CP57AC 44445851 IC50 = 16 nM T02752 CV6A2C 44445853 IC50 = 44 nM T02752 C6C1DS 44445854 IC50 = 0.9 nM T02752 CY0JI9 44445855 IC50 = 2.9 nM T02752 CLB89R 44445856 IC50 = 2 nM T02752 C53WTR 44445859 IC50 = 2.3 nM T02752 C1BVA3 44445861 IC50 = 3.3 nM T02752 C2BX1W 44445862 IC50 = 3.2 nM T02752 CQRN92 44445863 IC50 = 0.9 nM T02752 C4SA7D 44445864 IC50 = 1.5 nM T02752 CFZ8R7 44445865 IC50 = 0.7 nM T02752 COXK37 44445866 IC50 = 1.6 nM T02752 COK20T 44445867 IC50 = 1.3 nM T02752 CHX93V 44445868 IC50 = 0.9 nM T02752 CNM14B 44445870 IC50 = 1.3 nM T02752 C05MCY 44445872 IC50 = 0.9 nM T02752 C8X3DF 44445873 IC50 = 1.8 nM T02752 C76VUI 44445874 IC50 = 4 nM T02752 CXH5Z0 44445875 IC50 = 2.3 nM T02752 C5P6QX 44445876 IC50 = 2 nM T02752 CB75CU 44445877 IC50 = 3.6 nM T02752 C8CKU0 44445878 IC50 = 2.1 nM T02752 C97UQC 44445879 IC50 = 4.9 nM T02752 CJFW14 44445880 IC50 = 2.1 nM T02752 CUC7P1 44445883 IC50 = 2.5 nM T02752 C1X3MD 44445884 IC50 = 1.3 nM T02752 CCHB32 44445885 IC50 = 1.1 nM T02752 CWB3K5 44445886 IC50 = 0.6 nM T02752 C56YMC 44445887 IC50 = 1.6 nM T02752 C7PN6T 44445888 IC50 = 1.2 nM T02752 CS4XV5 44445889 IC50 = 2.6 nM T02752 CY2VI3 44445890 IC50 = 6.9 nM T02752 COF4U0 44445891 IC50 = 1.2 nM T02752 C1H8YR 44445892 IC50 = 2 nM T02752 C3C4DJ 44445893 IC50 = 2.7 nM T02752 CWZA43 44445894 IC50 = 2 nM T02752 C7XL0J 44445895 IC50 = 1.4 nM T02752 C3RZY0 44445896 IC50 = 2.8 nM T02752 C30QBA 44445901 IC50 = 1.2 nM T02752 C01JRH 44445907 IC50 = 2.5 nM T02752 CR19SE 44445915 IC50 = 1.2 nM T02752 C61XVE 44445916 IC50 = 1.5 nM T02752 C0OD2K 44447135 IC50 = 0.4 nM T02752 CDEX70 44447136 IC50 = 0.2 nM T02752 CZBN14 44447137 IC50 = 0.2 nM T02752 C3G8RI 44447138 IC50 = 0.4 nM T02752 CFUT83 44447139 IC50 = 0.4 nM T02752 C5OV4J 44447140 IC50 = 2.5 nM T02752 CYXP60 44447141 IC50 = 59 nM T02752 C69COR 44447142 IC50 = 421 nM T02752 CCWM93 44447143 IC50 = 0.3 nM T02752 CWE28C 44447144 IC50 = 2.6 nM T02752 C7Q0IM 44447145 IC50 = 0.5 nM T02752 CJ09DL 44447146 IC50 = 0.6 nM T02752 C05PSK 44447147 IC50 = 0.6 nM T02752 CWGB31 44447149 IC50 = 3.2 nM T02752 C48PKZ 44447150 IC50 = 9 nM T02752 CF96GA 44447153 IC50 = 211 nM T02752 CRP3N5 44447154 IC50 = 2.5 nM T02752 C73OVT 44447155 IC50 = 6 nM T02752 C2XCI0 44447161 IC50 = 21.6 nM T02752 C1L8EO 44447361 IC50 = 0.4 nM T02752 CUF2G5 44447366 IC50 = 577 nM T02752 CN4C7R 44447369 IC50 = 5.7 nM T02752 C16YFX 44447373 IC50 = 238 nM T02752 C7M5AT 44447374 IC50 = 19 nM T02752 CXI3J6 44447375 IC50 = 1.2 nM T02752 C2W5AE 44447377 IC50 = 88 nM T02752 CAK8W1 44447378 IC50 = 3.4 nM T02752 CFX7B9 44447380 IC50 = 2.5 nM T02752 CUV2C7 44447381 IC50 = 0.2 nM T02752 CXI13Y 44447382 IC50 = 0.004 nM T02752 C6IGQ5 44451928 IC50 = 38 nM T02752 C8DQ0E 44451981 IC50 = 1100 nM T02752 CVBE70 44451983 IC50 = 95 nM T02752 C6AFT4 44452009 IC50 = 2400 nM T02752 CGX8H6 44452044 IC50 = 3500 nM T02752 CVKW61 44452083 IC50 = 720 nM T02752 C9IT6Q 44452086 IC50 = 640 nM T02752 CPXO20 44452119 IC50 = 2900 nM T02752 C4K0XZ 44452120 IC50 = 670 nM T02752 C35WIN 44452168 IC50 = 20 nM T02752 CSBO17 44452172 IC50 = 4800 nM T02752 CBF8E9 44452198 IC50 = 9700 nM T02752 C3QWU9 44452220 IC50 = 2800 nM T02752 C7BVU5 44452248 IC50 = 810 nM T02752 C09KVL 44452250 IC50 = 1700 nM T02752 C60IWG 44452280 IC50 = 830 nM T02752 CO1RI7 44452304 IC50 = 600 nM T02752 CWEP85 44452361 IC50 = 3400 nM T02752 CC87TA 44455458 IC50 = 0.1 nM T02752 C68MTP 44455459 IC50 = 0.2 nM T02752 CN1U6E 44455460 IC50 = 2.7 nM T02752 C0V4OX 44455461 IC50 < 0.1 nM T02752 CDK31X 44455482 IC50 = 1.4 nM T02752 CI0K4G 44455483 IC50 = 0.304 nM T02752 C8WZB6 44455484 IC50 = 0.3 nM T02752 CYFI71 44455485 IC50 = 0.021 nM T02752 CZE05M 44455509 IC50 = 0.02 nM T02752 CMS92F 44455510 IC50 < 0.03 nM T02752 CN60DZ 44455511 IC50 = 1 nM T02752 C6OPJ8 44455539 IC50 = 1.1 nM T02752 C7O0AS 44455560 IC50 = 2 nM T02752 C4GOE6 44455625 IC50 = 0.8 nM T02752 CW1B8D 44455658 IC50 = 0.3 nM T02752 CX0B5K 44455683 IC50 = 0.05 nM T02752 CTV5H2 44455686 IC50 = 0.02 nM T02752 C2F6XP 44455711 IC50 = 0.013 nM T02752 CHCU69 44455744 IC50 < 0.03 nM T02752 CA6L8Y 44455745 IC50 = 0.05 nM T02752 CH67DO 44455765 IC50 = 1.7 nM T02752 CVH5R0 44455766 IC50 = 1.8 nM T02752 CD5U7E 44455767 IC50 = 2.7 nM T02752 CMC9H4 44455788 IC50 < 0.03 nM T02752 CM3R2V 44455790 IC50 = 1.2 nM T02752 CCD6Q4 44455791 IC50 = 0.6 nM T02752 C71TBV 44455792 IC50 > 1 nM T02752 CYF74A 44455793 IC50 = 0.06 nM T02752 C2BML0 44455817 IC50 = 0.87 nM T02752 C53JVI 44455818 IC50 = 1.2 nM T02752 C8B0KA 44455820 IC50 = 0.011 nM T02752 CP3KW7 44455841 IC50 = 0.4 nM T02752 CQ2KX1 44455844 IC50 = 0.6 nM T02752 C0A6GB 44455845 IC50 = 0.1 nM T02752 C6T5ZS 44455846 IC50 = 0.1 nM T02752 CIVE78 44455847 IC50 = 1.6 nM T02752 CU6AX0 44455869 IC50 = 0.02 nM T02752 CN0JV1 44455871 IC50 = 1 nM T02752 C28WVU 44455872 IC50 = 60 nM T02752 C1ED8S 44512617 IC50 = 1 nM T02752 C4M9FH 44512619 IC50 = 23 nM T02752 CT5N4E 44555481 IC50 > 50000 nM T02752 CS9U6X 44560288 IC50 = 93.7 nM T02752 C1MDQ6 44570537 IC50 = 0.23 nM T02752 C4DK1I 44570581 IC50 = 2.1 nM T02752 CJX87H 44570582 IC50 = 9.2 nM T02752 CAP51K 44570583 IC50 = 0.12 nM T02752 C1W9AF 44570584 IC50 = 0.15 nM T02752 CI1ZL9 44570617 IC50 = 1.1 nM T02752 C0OD7H 44570714 IC50 = 27.2 nM T02752 C3ZI2Y 44593546 IC50 = 5.5 nM T02752 C6PEV1 44593547 IC50 = 0.18 nM T02752 C0IE3Y 44593553 IC50 = 0.37 nM T02752 CTY83R 44593555 IC50 = 7 nM T02752 C2FVX5 45267588 IC50 = 0.98 nM T02752 CSWA06 45267629 IC50 = 140 nM T02752 CH5BI9 45268444 IC50 = 210 nM T02752 C2I1ZN 45268458 IC50 = 38 nM T02752 CE41PT 45268462 IC50 = 3.3 nM T02752 CT5E6A 45268467 IC50 = 6 nM T02752 CIRK70 45268519 IC50 = 320 nM T02752 CQJ6K5 45269291 IC50 = 250 nM T02752 CMU85W 45269302 IC50 = 3.6 nM T02752 CVZ1A3 45269320 IC50 = 7.5 nM T02752 CG8PH4 45269385 IC50 = 2500 nM T02752 C1VXZ6 45269392 IC50 = 100 nM T02752 C35LOA 45270135 IC50 = 2000 nM T02752 C57TQW 45270199 IC50 = 23 nM T02752 C1PSR2 45270977 IC50 = 160 nM T02752 CG4VI9 45270978 IC50 = 12 nM T02752 CJ7DN1 45270980 IC50 = 22 nM T02752 C1V6UG 45271843 IC50 = 14 nM T02752 CVD40I 45271882 IC50 = 230 nM T02752 CF32TD 45271891 IC50 = 1.8 nM T02752 C96EUD 45271892 IC50 = 1.6 nM T02752 CF6RA1 45271905 IC50 = 550 nM T02752 CX9Y5Q 45271911 IC50 = 170 nM T02752 CHMG80 45272697 IC50 = 5.1 nM T02752 CG10HX 45273619 IC50 = 900 nM T02752 C0M5IV 45273624 IC50 = 4.8 nM T02752 CY5LV6 45273632 IC50 = 5 nM T02752 CH97PL 45273639 IC50 = 45 nM T02752 CSB3T6 45273689 IC50 = 5.8 nM T02752 CP06XB 45273698 IC50 = 5.1 nM T02752 C6B5CT 45273705 IC50 = 300 nM T02752 CK59VA 57392726 IC50 = 1190 nM T02752 CJ3YB2 57394442 IC50 = 76 nM T02752 C2LX9H 57398008 IC50 = 82 nM T02752 C1N8YX 57401421 IC50 = 1000 nM T02752 C8K7EG 57718829 Ki = 38 nM T02752 CJXM43 57718837 Ki = 5.7 nM T02752 C90EAP 59295914 Ki = 12.59 nM T02752 CFX9H8 59295925 Ki = 7.943 nM T02752 C5P6UI 59295926 Ki = 12.59 nM T02752 C18YQX 59295928 Ki = 1 nM T02752 C9NMZ2 59295931 Ki = 1.585 nM T02752 CV6PS4 59295935 Ki = 1.995 nM T02752 CA8T3Q 59295938 Ki = 1.259 nM T02752 C59QBR 59295939 Ki = 2.512 nM T02752 COG4S6 59295946 Ki = 10 nM T02752 CHP65R 59295958 Ki = 3.162 nM T02752 CRNJ03 59295960 Ki = 19.95 nM T02752 C3PCY5 59295968 Ki = 0.7943 nM T02752 CYG56K 59295969 Ki = 3.981 nM T02752 C4PYU5 59295974 Ki = 2.512 nM T02752 CRZN12 59295978 Ki = 1.995 nM T02752 CR2T5D 59295982 Ki = 25.12 nM T02752 C4P3DW 59295984 Ki = 3.981 nM T02752 C17USX 59295994 Ki = 7.943 nM T02752 CJV58T 59296000 Ki = 2.512 nM T02752 C2K1TV 59296010 Ki = 1.585 nM T02752 C0KM5W 59296024 Ki = 6.31 nM T02752 CE73NG 59296033 Ki = 0.7943 nM T02752 CT2P4Z 59296039 Ki = 3.981 nM T02752 C21AHO 59296041 Ki = 63.1 nM T02752 CXK7O5 59296048 Ki = 3.981 nM T02752 CF53RX 59296064 Ki = 19.95 nM T02752 CPE0B2 59296066 Ki = 1.995 nM T02752 C07OPL 59296073 Ki = 158.49 nM T02752 CFR8S7 59296077 Ki = 15.85 nM T02752 CMD56H 59296081 Ki = 0.3162 nM T02752 C2HP9B 59296085 Ki = 251.19 nM T02752 CFCE90 59296090 Ki = 3.162 nM T02752 CGIL10 59296094 Ki = 3.981 nM T02752 C4H8KW 59296098 Ki = 31.62 nM T02752 CUC57E 59296099 Ki = 0.7943 nM T02752 C1ZN0M 59296100 Ki = 3.162 nM T02752 CX6JS1 59296104 Ki = 2.512 nM T02752 CZW0V1 59296109 Ki = 15.85 nM T02752 C5TMB2 59296111 Ki = 6.31 nM T02752 CGF80H 59296114 Ki = 199.53 nM T02752 CECR98 66615606 Ki = 1.259 nM T02752 CJ85YZ 66615617 Ki = 1.995 nM T02752 C9IQ1Y 66615619 Ki = 0.5012 nM T02752 CFO03A 66615627 Ki = 0.1995 nM T02752 CA59FS 66615678 Ki = 3.981 nM T02752 C9P6ZL 66615691 Ki = 1.585 nM T02752 C75RXH 66615702 Ki = 0.7943 nM T02752 CL69HQ 66615705 Ki = 5.012 nM T02752 CA8I4E 66906657 Ki = 31 nM T02752 CHN01B 68826395 IC50 = 7.4 nM T02752 C6FZD0 68846936 Ki = 79.43 nM T02752 CZPM30 68849581 Ki = 31.62 nM T02752 C5PY2V 68938028 Ki = 5.012 nM T02752 C07YOG 69260079 Ki = 630.96 nM T02752 CV7P3D 69260851 Ki = 158.49 nM T02752 C4QO7E 69260946 Ki = 100 nM T02752 CO9U3M 69262172 Ki = 1.995 nM T02752 C7HN5L 69272932 Ki = 31.62 nM T02752 CJ2D3I 69274365 Ki = 39.81 nM T02752 COD5Y1 69347575 Ki = 10 nM T02752 C51DQR 69347707 Ki = 630.96 nM T02752 C8F1CY 69347719 Ki = 19.95 nM T02752 C93COF 69347980 Ki = 251.19 nM T02752 CPW42A 69348078 Ki = 31.62 nM T02752 CZO27L 69826668 Ki = 5.012 nM T02752 CZ49WC 70682098 IC50 = 44 nM T02752 C1FD8W 70682099 IC50 = 310 nM T02752 CD7F8P 70682100 IC50 = 1600 nM T02752 C87GBP 70682101 IC50 = 440 nM T02752 CS3GQ5 70682102 IC50 = 13 nM T02752 C25LIT 70684221 IC50 = 780 nM T02752 CUD96V 70684230 IC50 = 31 nM T02752 C1KV4D 70686357 IC50 = 380 nM T02752 C7TRV3 70686358 IC50 = 13 nM T02752 CP1A5W 70688459 IC50 = 18 nM T02752 C7DP3F 70688460 IC50 = 920 nM T02752 CQ6J4D 70688469 IC50 = 29 nM T02752 CO12FZ 70688470 IC50 = 30 nM T02752 C7BW8F 70690517 IC50 = 59 nM T02752 CH7GX0 70690518 IC50 = 360 nM T02752 CK0F6M 70690519 IC50 = 52 nM T02752 C9O5EX 70690520 IC50 = 56 nM T02752 CGF2J9 70692659 IC50 = 190 nM T02752 C49NKO 70692666 IC50 = 45 nM T02752 C1A6KV 70694701 IC50 = 62 nM T02752 C67KAT 70694702 IC50 = 51 nM T02752 CB78WS 70694703 IC50 = 110 nM T02752 C2M4AE 70696744 IC50 = 20 nM T02752 CV2RZ5 70696751 IC50 = 8 nM T02752 C1YP3E 70696752 IC50 = 63 nM T02752 C6GN5H 70696753 IC50 = 240 nM T02752 C4YE5N 70696765 IC50 = 4.9 nM T02752 C18RLK 71072034 Ki = 31.62 nM T02752 C4C0SP 71072040 Ki = 10 nM T02752 C1YNH6 71072044 Ki = 10 nM T02752 CVU3G7 71072050 Ki = 10 nM T02752 C2M1JY 71072052 Ki = 7.943 nM T02752 CE6Y8Z 71072057 Ki = 25.12 nM T02752 C0Z3KN 71072081 Ki = 19.95 nM T02752 C3FR6X 71072104 Ki = 3.981 nM T02752 C1BEC9 71072113 Ki = 19.95 nM T02752 CNY09L 71072115 Ki = 19.95 nM T02752 CFNZ23 71072118 Ki = 10 nM T02752 CTNZ18 71449114 IC50 = 28 nM T02752 CH5X6M 71449584 Ki = 19.95 nM T02752 CH5PX8 71449585 Ki = 39.81 nM T02752 CGE2I8 71449677 IC50 = 14 nM T02752 C45XDF 71449694 IC50 = 110 nM T02752 C0O2JU 71449695 IC50 = 600 nM T02752 CUKW48 71449857 Ki = 251.19 nM T02752 COVR94 71449858 Ki = 79.43 nM T02752 C5M7WE 71449859 Ki = 398.11 nM T02752 CSYN25 71450777 Ki = 794.33 nM T02752 C3FC1H 71451390 Ki = 50.12 nM T02752 C4W6YG 71451391 Ki = 12.59 nM T02752 CI65MW 71451392 Ki = 3.162 nM T02752 C25NZT 71451489 IC50 = 9.9 nM T02752 C68UFH 71451670 Ki = 5011.87 nM T02752 C9OG2Q 71451671 Ki = 501.19 nM T02752 CE1Z0V 71452601 Ki = 31.62 nM T02752 C59WFT 71452602 Ki = 316.23 nM T02752 C8C9JT 71453204 Ki = 7.943 nM T02752 C56NWY 71453334 IC50 = 23 nM T02752 CHM82W 71453335 IC50 = 50 nM T02752 CJ3W6B 71453336 IC50 = 44 nM T02752 C5SQO7 71453337 IC50 = 25 nM T02752 CB86VX 71453505 Ki = 31.62 nM T02752 C02FKR 71454296 Ki = 3.981 nM T02752 CZ8W9G 71454365 Ki = 158.49 nM T02752 C2EFA4 71454583 IC50 = 802 nM T02752 CIT10B 71455028 IC50 = 50 nM T02752 C5E7XW 71455029 IC50 = 24 nM T02752 CQ41KH 71455044 IC50 = 44 nM T02752 CB6PF0 71455217 Ki = 125.89 nM T02752 CL9BS3 71456722 Ki = 1.995 nM T02752 CT0OQ6 71456725 Ki = 25.12 nM T02752 CVYG02 71456816 IC50 = 44 nM T02752 CKR3H0 71456839 IC50 = 28 nM T02752 CHQM97 71456840 IC50 = 71 nM T02752 CIXY68 71457009 Ki = 630.96 nM T02752 CGP6K8 71457010 Ki = 5.012 nM T02752 C7ML3X 71458114 IC50 = 169 nM T02752 CP9SM0 71458677 IC50 = 12 nM T02752 CZW7X0 71458868 Ki = 3.162 nM T02752 CHC0Z2 71458869 Ki = 251.19 nM T02752 CF1PV0 71458870 Ki = 2511.89 nM T02752 CJ1M6I 71459762 Ki = 1.585 nM T02752 CMI1A6 71459825 Ki = 125.89 nM T02752 CP26GF 71460416 Ki = 25.12 nM T02752 CH51UB 71460419 Ki = 19.95 nM T02752 CF50RP 71460504 IC50 = 41 nM T02752 CZ8J6L 71460523 IC50 = 0.87 nM T02752 CELP64 71460524 IC50 = 380 nM T02752 CZY57V 71460525 IC50 = 2.4 nM T02752 C1GV6P 71461541 Ki = 79.43 nM T02752 C9UG2X 71462100 Ki = 1.259 nM T02752 CYM4X2 71462102 Ki = 125.89 nM T02752 CL4MZ5 71462103 Ki = 100 nM T02752 CL2TK1 71462226 IC50 = 51 nM T02752 C30WJF 71462227 IC50 = 2000 nM T02752 CX97KJ 71462389 Ki = 199.53 nM T02752 C6UBQ4 71462390 Ki = 199.53 nM T02752 CQ36LR 71462391 Ki = 398.11 nM T02752 C5CS7I 71463287 Ki = 251.19 nM T02752 C05HIC 71463288 Ki = 125.89 nM T02752 CM9B0T 76309741 IC50 = 131 nM T02752 C1UOY7 76313414 IC50 = 93 nM T02752 C8RM5L 76313428 IC50 = 29 nM T02752 CXC2S5 76313429 IC50 = 679 nM T02752 CTN57W 76313430 IC50 = 85 nM T02752 C6FX7K 76316938 IC50 = 23 nM T02752 CT37MX 76316939 IC50 = 12 nM T02752 C2S8OX 76316987 IC50 = 29 nM T02752 C1QL8W 76320667 IC50 = 613 nM T02752 C6YW3I 76320668 IC50 = 89 nM T02752 C4G0CX 76320669 IC50 = 98 nM T02752 C1JK9P 76320670 IC50 = 217 nM T02752 CJ5F3N 76320671 IC50 = 279 nM T02752 CT2D5P 76320703 IC50 = 3500 nM T02752 CYMO73 76324312 IC50 = 482 nM T02752 CC8JI7 76324313 IC50 = 57 nM T02752 CEAQ91 76327878 IC50 = 13 nM T02752 CGO16S 76327879 IC50 = 44 nM T02752 CZE1O7 76327880 IC50 = 225 nM T02752 C9JV4B 76331526 IC50 = 221 nM T02752 C7Q8YI 76331527 IC50 = 118 nM T02752 C6ENV5 100951623 EC50 > 10000 nM T02752 C9SV0C 118721184 Ki = 60 nM T02752 CW45XR 118721185 Ki = 32 nM T02752 CR6JB3 118721186 Ki = 78 nM T02752 CL3P7T 118721187 Ki = 96 nM T02752 C4BG3Z 118721188 Ki = 450 nM T02752 CDXP86 118721189 Ki = 33 nM T02752 CS62YE 118721190 Ki = 99 nM T02752 C9IWE7 118721191 Ki = 4.3 nM T02752 C2WC7G 118721192 Ki = 480 nM T02752 C2UPR3 118721193 Ki = 66 nM T02752 C7IX5C 118721194 Ki = 4.8 nM T02752 C53ZRD 118721195 Ki = 46 nM T02752 CBZR06 118721196 Ki = 86 nM T02752 C8E0NK 118721197 Ki = 190 nM T02752 CXLM39 118721198 Ki = 310 nM T02752 C6R1ME 118721199 Ki = 4000 nM T02752 CC04YW 118721200 Ki = 4.7 nM T02752 CJ4HE3 118721201 Ki = 6900 nM T02752 CC28BD 118721202 Ki = 5 nM T02752 CQCX23 118721203 Ki = 98 nM T02752 C7C3DB 118721204 Ki = 11 nM T02752 CR30ZQ 118721205 Ki = 4 nM T02752 CY89CH 118721206 Ki = 34 nM T02752 CM6R5Q 124396489 EC50 = 1600 nM T02752 C0KVF7 136216709 Ki = 830 nM T02752 C78RFZ 136229178 Ki = 316.23 nM T02752 D01JZV 9913085 IC50 = 2.3 nM T09130 D01AZG 5073 Ki > 5000 nM T09130 D05DVP 5717 IC50 > 10000 nM T09130 D07ZTO 2370 Ki = 97 nM T09130 D0D1AL 3559 Ki = 4670 nM T09130 D0H7KF 5002 Ki = 1020 nM T09130 D0O2WB 4991 Ki > 100000 nM T09130 D0R1JV 60854 Ki > 5000 nM T09130 D0RG3O 174174 Ki = 0.32 nM T09130 D0T0LM 4848 Ki = 530 nM T09130 D0U7BW 5831 EC50 = 100 nM T09130 D0V4QS 135398745 Ki = 26 nM T09130 D0Z1RV 135398737 Ki = 34 nM T09130 D07EFM 2230 EC50 = 73 nM T09130 D0A7KI 3037308 Ki = 1130 nM T09130 D0O2XQ 11256587 IC50 > 17000 nM T09130 D00OWF 5280953 Ki > 10000 nM T09130 D08AWI 11430856 Ki > 2000 nM T09130 D0OS6O 60149 Ki > 5000 nM T09130 C45PUM 2551 Ki = 5 nM T09130 C9IK1Y 4136 Ki = 150 nM T09130 CL9I7S 19716 Ki = 4960 nM T09130 CM6TE9 55005 Ki = 330 nM T09130 C0AMN5 84607 Ki = 1200 nM T09130 C27RUO 129486 Ki = 0.27 nM T09130 CGT8R0 160510 Ki > 10000 nM T09130 CZ0UI5 208598 Ki = 28000 nM T09130 CYV1R3 417052 Ki > 10000 nM T09130 CF23YW 535891 Ki = 6700 nM T09130 CJ94ZR 578008 Ki = 10900 nM T09130 CFR90P 578009 Ki = 4900 nM T09130 CE4KC8 3038603 Ki = 4.3 nM T09130 C54FEG 3039881 Ki = 43 nM T09130 CCNJ91 9794960 Ki = 2.8 nM T09130 CJ8LT7 9848518 IC50 > 10000 nM T09130 CGO07X 9859365 Ki = 9.6 nM T09130 CT2C6K 9870702 IC50 > 10000 nM T09130 CL1OJ6 9972276 Ki = 39 nM T09130 CD9A5M 9991939 Ki = 550 nM T09130 C8F4XT 9991979 Ki = 760 nM T09130 C2WJS1 10058649 Ki = 920 nM T09130 CV6A5I 10061123 Ki = 5400 nM T09130 CT4XE6 10103909 Ki = 6100 nM T09130 CHUE04 10104527 Ki > 38000 nM T09130 COR41M 10105880 Ki = 19000 nM T09130 CE69PK 10242813 Ki = 580 nM T09130 CQB1O6 10243426 Ki = 240 nM T09130 CEYJ57 10244370 Ki = 8100 nM T09130 CWP67J 10330721 Ki = 45000 nM T09130 CLW9R8 10330893 Ki = 870 nM T09130 C9YR5B 10339062 Ki = 2000 nM T09130 C5M9WO 10354430 Ki = 6900 nM T09130 CUBA69 10398843 Ki = 310 nM T09130 C3C7SG 10425107 Ki = 15 nM T09130 C07QHE 10429011 Ki = 600 nM T09130 CI8R9A 10465050 Ki = 3700 nM T09130 CK9ZH7 10466231 Ki = 120 nM T09130 CVK48E 10467755 Ki = 8600 nM T09130 C53SCK 10468535 Ki = 249 nM T09130 C26BIM 10475156 Ki = 20000 nM T09130 CE49XD 10482127 Ki = 4700 nM T09130 C64MHO 10488962 Ki = 1300 nM T09130 CJUZ01 10489806 Ki = 1100 nM T09130 CN61QO 10491094 Ki = 364 nM T09130 CF26AB 10491129 Ki = 6.4 nM T09130 CMJH27 10491230 Ki = 1400 nM T09130 C24TYJ 10494696 Ki = 40 nM T09130 COZ04I 10515035 Ki = 648 nM T09130 C65JQC 10519655 Ki = 130 nM T09130 CIPS94 10520427 Ki = 1.55 nM T09130 C2E9OY 10540939 Ki = 1170 nM T09130 CUJ54L 10542335 Ki = 20 nM T09130 CH2IN4 10544852 Ki = 420 nM T09130 C8X4GK 10547508 Ki = 440 nM T09130 CC90SN 10559551 Ki = 12 nM T09130 CW6N1F 10560716 Ki = 570 nM T09130 CW70HG 10561983 Ki = 25 nM T09130 CSPV18 10562031 Ki = 212 nM T09130 CL5PA0 10564410 Ki = 7.8 nM T09130 CMH3Y1 10566215 Ki = 135 nM T09130 C3O7WR 10567945 Ki = 8.4 nM T09130 CJUI84 10595980 Ki = 197 nM T09130 C39YPC 10609662 Ki = 60 nM T09130 C4GDM6 10620744 Ki > 150 nM T09130 C8FJN1 10631505 Ki = 520 nM T09130 C1CGR8 10635414 Ki = 2.39 nM T09130 CYTX65 10638038 Ki = 289 nM T09130 C9LJ4N 10639323 Ki = 5.7 nM T09130 CGF7H3 10657635 Ki = 25.3 nM T09130 CMDJ73 10657636 Ki = 116 nM T09130 C3GX5N 10657853 Ki = 6.3 nM T09130 C3CW5S 10658329 Ki = 60 nM T09130 CHS6V7 10658402 Ki = 730 nM T09130 CN3M6E 10660333 Ki = 38 nM T09130 C0O4NE 10660795 Ki = 3665 nM T09130 CUEM15 10668605 Ki = 16 nM T09130 C51YMH 10679529 Ki = 400 nM T09130 CJX70U 10679530 Ki = 710 nM T09130 C6G1HZ 10679666 Ki = 7.4 nM T09130 C1CF6K 10683266 Ki = 0.27 nM T09130 CB1E8Q 10685209 Ki = 3320 nM T09130 C3XYU9 10691101 Ki = 314 nM T09130 C5UBV6 10706187 Ki = 330 nM T09130 CG4OS3 10707802 Ki = 1.9 nM T09130 CO7V2I 10711058 Ki = 280 nM T09130 C8XH4J 10729440 Ki = 330 nM T09130 C85KEU 10731181 Ki = 190 nM T09130 C18FGL 10736293 Ki = 8.2 nM T09130 CBM28Y 10751241 Ki = 1100 nM T09130 C3H0PJ 10754304 Ki = 0.79 nM T09130 CLKQ97 10754495 Ki = 139 nM T09130 CA8WB1 10757263 Ki = 2.2 nM T09130 CY69KE 10774406 Ki = 93 nM T09130 CQ6NP7 10775987 Ki = 810 nM T09130 C93RXU 10809840 Ki = 480 nM T09130 C6O7HR 10823129 Ki = 21 nM T09130 C5OZ2M 10824792 Ki = 130 nM T09130 CDH5S7 10827641 Ki = 800 nM T09130 CK4LY6 10827642 Ki = 220 nM T09130 CC69TA 10830695 Ki = 2.3 nM T09130 CJ52AK 10833559 Ki = 221 nM T09130 C0RKE3 10847131 Ki = 17.1 nM T09130 CTP7C4 10848516 Ki = 140 nM T09130 C5J3KH 10903857 Ki > 100000 nM T09130 CM21SA 10982024 Ki = 29000 nM T09130 CVT4O0 11014962 Ki = 42000.1 nM T09130 CM16PV 11034977 Ki = 75000.1 nM T09130 C48WOS 11069873 Ki = 8100.01 nM T09130 CIG85H 11282247 IC50 > 5500 nM T09130 C5M3ZN 11329138 IC50 > 33000 nM T09130 C3MQW7 11819545 Ki = 4300 nM T09130 C0BPK3 11819882 Ki = 290 nM T09130 C2KW3U 11819883 Ki = 3700 nM T09130 C7E5PA 11826864 Ki = 2600 nM T09130 CXLW54 11948707 Ki > 10000 nM T09130 CKY94S 12866543 Ki = 940 nM T09130 CWP60M 13621534 IC50 > 50000 nM T09130 C7NL5D 13621548 IC50 = 35000 nM T09130 C8GDT6 13621550 IC50 > 50000 nM T09130 CEGU40 13621552 IC50 = 11000 nM T09130 C38UXQ 13621554 IC50 = 49000 nM T09130 CR91KI 13621558 IC50 > 50000 nM T09130 CTCX78 13621560 IC50 = 48000 nM T09130 C5PRZ0 13621564 IC50 = 22000 nM T09130 C0O8JQ 13621575 IC50 > 50000 nM T09130 CB65YF 14511183 Ki = 5600 nM T09130 C5KGZ4 14511184 Ki = 43000 nM T09130 CCT6Q8 14511186 Ki = 19600 nM T09130 CU36CN 14685523 Ki = 2400 nM T09130 C89WTN 14761795 EC50 = 2800 nM T09130 CN19PC 14801695 EC50 = 320 nM T09130 CPZ2U6 14801696 EC50 > 30000 nM T09130 C0RNI4 14801697 EC50 > 30000 nM T09130 CNCM93 14801698 EC50 > 30000 nM T09130 CE4MH3 14801702 EC50 > 30000 nM T09130 CY5I0K 14801703 EC50 > 30000 nM T09130 C4L0PS 15114748 Ki = 18000 nM T09130 CSA5Y2 15196231 Ki > 58000 nM T09130 CO4EB0 15196232 Ki = 24700 nM T09130 COIG73 15196233 Ki = 28000 nM T09130 C80ICP 15196234 Ki = 300 nM T09130 CIV27H 15196235 Ki = 11000 nM T09130 CXZB18 15196236 Ki = 410 nM T09130 CEH60Q 15196354 Ki = 3800 nM T09130 C12FIS 15599352 Ki = 0.054 nM T09130 CTSN15 15629545 EC50 = 7500 nM T09130 C6OGR3 18960834 EC50 = 720 nM T09130 CC7E1Z 18960880 EC50 > 30000 nM T09130 CW9S3A 18960891 EC50 = 1280 nM T09130 CPVY15 18960911 EC50 > 30000 nM T09130 C3IQT5 23352279 Ki = 2600 nM T09130 CD1H7X 23352282 Ki = 73 nM T09130 C5SUY3 23352285 Ki = 5700 nM T09130 C6Z3VB 44299828 IC50 > 100 nM T09130 C0PJ6Y 44299849 IC50 > 100 nM T09130 CR9C5F 44300131 IC50 > 100 nM T09130 CYGT05 44300167 IC50 > 100 nM T09130 C29NZB 44300171 IC50 > 100 nM T09130 C4O0YB 44300172 IC50 > 100 nM T09130 CVCF79 44300182 IC50 > 100 nM T09130 CDA0F8 44300196 IC50 > 100 nM T09130 C0T2WP 44300224 IC50 > 100 nM T09130 C9HJ7T 44300228 IC50 > 100 nM T09130 CK17EG 44300229 IC50 > 100 nM T09130 CR6Y8E 44300230 IC50 > 100 nM T09130 CS9AY0 44300232 IC50 > 100 nM T09130 CSB2C6 44300238 IC50 > 100 nM T09130 CB4M8W 44300239 IC50 > 100 nM T09130 C7XMU4 44300240 IC50 > 100 nM T09130 C89CIB 44300243 IC50 > 100 nM T09130 CSE35C 44328347 Ki = 8000 nM T09130 CM6D4U 44328348 Ki > 5000 nM T09130 C8O4PB 44328540 Ki = 2500 nM T09130 CP5W3M 44328561 Ki = 1900 nM T09130 CP53TO 44337748 Ki = 4190 nM T09130 C8EGW9 44337753 Ki = 0.475 nM T09130 C21ILP 44337760 Ki = 19.1 nM T09130 C9BX7V 44337761 Ki = 9.64 nM T09130 CR0BL8 44337776 Ki = 4570 nM T09130 C5LA3S 44348983 Ki = 99 nM T09130 C3DO4B 44349519 Ki = 0.8 nM T09130 CF8AP4 44374542 EC50 = 32 nM T09130 C8V9RH 44374587 EC50 > 30000 nM T09130 CS96DJ 44374588 EC50 > 30000 nM T09130 CG28OF 44374624 EC50 = 420 nM T09130 CER70L 44374625 EC50 > 30000 nM T09130 C5LEO9 44374635 EC50 = 1000 nM T09130 CT2H9K 44374651 EC50 > 30000 nM T09130 C1QF6W 44374652 EC50 = 150 nM T09130 C5IB6N 44374653 EC50 = 130 nM T09130 CS97DA 44374661 EC50 = 620 nM T09130 CQ46CL 44374678 EC50 > 30000 nM T09130 C7C6RT 44374689 EC50 > 30000 nM T09130 C7MXL8 44374694 EC50 = 1460 nM T09130 CLT21F 44374704 EC50 = 100 nM T09130 C1GZ9I 44374705 EC50 = 200 nM T09130 CZRH30 44374767 EC50 > 30000 nM T09130 C3ZY5W 44377401 Ki = 1400 nM T09130 C7YU9S 46878250 Ki = 7700 nM T09130 CU7OY8 54584893 EC50 = 94 nM T09130 CL45WN 57345320 IC50 > 14000 nM T09130 CDI84E 71450922 IC50 > 10000 nM T09130 CP0D2T 71454526 Ki = 3750 nM T09130 C2DP1L 135313576 IC50 = 28500 nM T09130 C76OJC 135313705 IC50 > 17000 nM T09130 CO4W2L 135313730 IC50 > 16700 nM T09130 CN7U0V 135313757 IC50 > 16700 nM T09130 C0G6IE 135313758 IC50 = 5900 nM T09130 CD5FU8 135313764 IC50 > 16700 nM T09130 C74VEJ 135313789 IC50 > 16700 nM T09130 CO7AJ2 135313829 IC50 = 4350 nM T09130 C10GDT 135313911 IC50 = 3000 nM T09130 CMR34P 135313919 IC50 > 17000 nM T09130 CJAQ57 135313931 IC50 = 11500 nM T09130 CQR2M1 135313955 IC50 > 16700 nM T09130 CS5HY9 135313960 IC50 = 6100 nM T09130 C9FNU5 135313965 IC50 > 17000 nM T09130 CQ4B1T 135313976 IC50 = 10700 nM T09130 CD8B0A 135313980 IC50 > 33000 nM T09130 CGPC70 135313983 IC50 > 33000 nM T09130 C75MZN 135314048 IC50 > 16700 nM T09130 CUA3M7 135314064 IC50 > 27000 nM T09130 CL12JU 135314107 IC50 = 11100 nM T09130 CPTO20 135314108 IC50 = 15400 nM T09130 C1XSQ4 135314132 IC50 = 33000 nM T09130 CFD5N1 135314164 IC50 > 21000 nM T09130 C63BWA 135314215 IC50 = 23200 nM T09130 C57HTM 135314218 IC50 = 11630 nM T09130 CU67EM 135314256 IC50 > 16700 nM T09130 CL23RS 135314305 IC50 > 33000 nM T09130 CMC3E1 135314326 IC50 > 16700 nM T09130 CWI13E 135314362 IC50 = 9560 nM T09130 CL6FK9 135314383 IC50 > 33000 nM T09130 C5OU1T 135409492 Ki = 662 nM T09130 C4PM9W 135515431 Ki = 501 nM T09130 CYDF05 142416702 IC50 > 33000 nM T09130 C06ZBJ 142416740 IC50 > 16700 nM T09130 CZA08U 142416759 IC50 > 33000 nM T09130 C7C3MK 142416935 IC50 > 16700 nM T09130 CVND41 145949156 IC50 > 17000 nM T09130 CI14LP 145949343 IC50 > 14000 nM T09130 C8KA6P 145949486 IC50 = 3200 nM T09130 CA0B3D 145949907 IC50 > 33300 nM T09130 C7W9ZT 145949949 IC50 = 8340 nM T09130 CAT5E1 145950272 IC50 > 16700 nM T09130 CAWU95 145950510 IC50 > 16700 nM T09130 CL2OR1 145950976 IC50 = 7180 nM T09130 C2M8PI 145951236 IC50 > 16700 nM T09130 CC4K9F 145952601 IC50 > 17000 nM T09130 CGW92C 145952721 IC50 > 14000 nM T09130 C2FXL5 145952723 IC50 = 887 nM T09130 CER83S 145953040 IC50 = 8600 nM T09130 C1A4CH 145953177 IC50 > 33300 nM T09130 COZ1F4 145953325 IC50 = 26300 nM T09130 C09WNF 145953342 IC50 > 14000 nM T09130 CEJ26X 145953403 IC50 > 17000 nM T09130 CS21ZB 145953739 IC50 > 17000 nM T09130 C59AVT 145954818 IC50 > 33300 nM T09130 C4P6MT 145954878 IC50 = 1980 nM T09130 CK0S1G 145955694 IC50 > 17000 nM T09130 CE03RK 145955745 IC50 > 33300 nM T09130 CF6T7G 145955884 IC50 = 21600 nM T09130 C8Y4VT 145956312 IC50 = 15100 nM T09130 CXAR52 145956817 IC50 > 16700 nM T09130 CQ0JP4 145957239 IC50 = 2100 nM T09130 CK94HO 145957365 IC50 > 14000 nM T09130 C70LMY 145957553 IC50 > 33300 nM T09130 CB2K0W 145957599 IC50 = 10800 nM T09130 C8WZY3 145958093 IC50 > 14000 nM T09130 C3TX8O 145958528 IC50 > 14000 nM T09130 CT3U1A 145958698 IC50 = 9250 nM T09130 CW8M0I 145959142 IC50 > 33300 nM T09130 C8DH5F 145959814 IC50 > 14000 nM T09130 C5Z9US 145959844 IC50 = 6560 nM T09130 CUD9E6 145960079 IC50 = 17900 nM T09130 C3F8XM 145960247 IC50 > 16700 nM T09130 CD01PX 145961863 IC50 = 4980 nM T09130 C64OLM 145963140 IC50 = 26100 nM T09130 CU8Y2C 145963537 IC50 > 17000 nM T09130 CND2K7 145971189 IC50 > 17000 nM T09130 CMI45E 145971507 IC50 = 3160 nM T09130 CP7LW2 145973146 IC50 > 33300 nM T09130 C8OSM0 145973345 IC50 > 16700 nM T09130 C54QHK 145974080 IC50 = 5600 nM T09130 CP20BX 145974804 IC50 > 16700 nM T09130 CP9TR0 10324985 Ki > 10000 nM T09130 CJU8R4 14737773 Ki = 10400 nM T09130 C4NB3O 15108132 Ki = 8.21 nM T09130 CW4EQ2 15108134 Ki = 12.8 nM T09130 CX4HN3 15599354 Ki = 0.449 nM T09130 D00SDJ 11237664 IC50 > 10000 nM T09130 D02VGM 23056 Ki = 0.045 nM T09130 D05GDP 599482 Ki > 10000 nM T09130 D05KUM 135446209 Ki = 333 nM T09130 D0P1FJ 71128 Ki = 23 nM T51385 D0V1WQ 24857286 EC50 > 10000 nM T51385 C8AND5 7789 EC50 = 1737.8 nM T51385 CKRG59 10466 EC50 = 1698.24 nM T51385 CWY93I 37289 EC50 > 100000 nM T51385 CXH9K8 169433 EC50 > 100000 nM T51385 CF1W7M 233085 IC50 = 79.43 nM T51385 C7KQP3 258072 EC50 = 12589.25 nM T51385 CAP29L 272261 EC50 > 31622.78 nM T51385 CC05OD 561372 EC50 = 11748.98 nM T51385 C19ADF 643684 EC50 = 1318.26 nM T51385 CA9GQ6 674995 EC50 = 3548.13 nM T51385 CN38UP 711134 EC50 = 2511.89 nM T51385 CZN6S9 743974 EC50 = 489.78 nM T51385 CA3BW5 796476 EC50 > 31622.78 nM T51385 CU1B6N 825631 EC50 = 3162.28 nM T51385 CSP07R 834320 EC50 > 31622.78 nM T51385 C3EBU9 835355 EC50 > 31622.78 nM T51385 CJ5T4B 841618 EC50 = 3162.28 nM T51385 CFUM73 896519 EC50 > 31622.78 nM T51385 CX4NK5 900631 EC50 = 316.23 nM T51385 C0LCE8 925016 EC50 = 1000 nM T51385 C0TPC6 956298 EC50 = 3981.07 nM T51385 CL67RF 975397 EC50 = 10000 nM T51385 C0W7CJ 977153 EC50 = 794.33 nM T51385 CB53NT 2843133 EC50 = 5370.32 nM T51385 C60EVX 2906141 EC50 > 31622.78 nM T51385 CGH79K 3518281 EC50 = 6309.57 nM T51385 COT13S 5312743 EC50 > 100000 nM T51385 C7ASQ0 5312744 EC50 > 100000 nM T51385 CW5R4H 8190702 EC50 = 7943.28 nM T51385 CP03EA 8190712 EC50 = 398.11 nM T51385 CUL61X 8190724 EC50 = 1258.93 nM T51385 C43THE 8190727 EC50 = 1995.26 nM T51385 C6LMK5 8190733 EC50 > 31622.78 nM T51385 CNZ5W7 10176767 EC50 > 100000 nM T51385 CBJ23P 14454530 EC50 > 100000 nM T51385 CE3JI2 23136363 EC50 = 562.34 nM T51385 CV2HD8 23136401 EC50 = 501.19 nM T51385 CD4VG3 23136411 EC50 = 2398.83 nM T51385 CW3AM0 23136477 EC50 = 371.54 nM T51385 CTQ53W 23346507 EC50 = 57543.99 nM T51385 CIA3X8 23699039 EC50 > 100000 nM T51385 CY0F4L 24825484 EC50 = 58884.37 nM T51385 CHX09F 24825492 EC50 = 3090.3 nM T51385 C56XKE 24825509 EC50 = 4466.84 nM T51385 CS8T2B 25109512 EC50 = 1700 nM T51385 CZ39BV 25149901 EC50 = 8511.38 nM T51385 CZ7U2W 46869922 EC50 > 10000 nM T51385 CYTP35 46892131 EC50 = 181.97 nM T51385 CB86TC 46908122 EC50 = 5011.87 nM T51385 CP9JN0 51349861 EC50 = 16595.87 nM T51385 CAS51V 51350138 EC50 = 8317.64 nM T51385 C4EGI3 51350272 EC50 = 8709.64 nM T51385 C7AI4W 54580132 EC50 = 1737.8 nM T51385 CS03YA 54582149 EC50 = 20892.96 nM T51385 CKV29F 54582150 EC50 = 51286.14 nM T51385 CU5K1Y 54583098 EC50 = 4786.3 nM T51385 C31NYG 54584098 EC50 = 478.63 nM T51385 CDYZ19 54585039 EC50 = 5370.32 nM T51385 C03CFM 54586011 EC50 = 1288.25 nM T51385 C2W0GK 54586984 EC50 = 6760.83 nM T51385 CZ1M3Q 54757519 EC50 > 100000 nM T51385 CY5O1Q 57521702 EC50 = 7079.46 nM T51385 CDW9N4 57521808 EC50 = 1949.84 nM T51385 CZL1W6 57521809 EC50 = 177.83 nM T51385 CT06GY 57521810 EC50 = 588.84 nM T51385 C9S5CH 57521811 EC50 = 309.03 nM T51385 C2DUX1 57521812 EC50 = 295.12 nM T51385 CD8G6M 57521813 EC50 = 2041.74 nM T51385 CDRW60 57521814 EC50 = 190.55 nM T51385 C76WSM 57521913 EC50 = 2187.76 nM T51385 C9O0LB 57521914 EC50 = 4365.16 nM T51385 CS6B7Q 57521915 EC50 = 234.42 nM T51385 CV8F2A 57521916 EC50 = 239.88 nM T51385 CBTP21 57521917 EC50 = 912.01 nM T51385 CPZQ75 57521918 EC50 = 512.86 nM T51385 CH9K1N 57521919 EC50 = 109.65 nM T51385 C68FGV 57839754 EC50 = 750 nM T51385 CA5X0H 59455552 EC50 = 610 nM T51385 C9XH0G 59455555 EC50 = 270 nM T51385 CI0NP9 59455584 EC50 = 520 nM T51385 CEOP18 60195036 EC50 = 10964.78 nM T51385 CR9C7I 60195038 EC50 = 8511.38 nM T51385 CX30BG 60195039 EC50 = 4265.8 nM T51385 C7S3HJ 60195040 EC50 = 93325.43 nM T51385 CQLD97 60195125 EC50 = 43651.58 nM T51385 C9DH3R 66562286 EC50 = 7943.28 nM T51385 C16SUO 66562287 EC50 > 100000 nM T51385 CB75OA 66562288 EC50 = 19952.62 nM T51385 CEK8U4 66562289 EC50 = 26302.68 nM T51385 C04XUT 66562385 EC50 = 1584.89 nM T51385 CI73FC 66562386 EC50 = 9549.93 nM T51385 CH5JZ6 66562387 EC50 > 100000 nM T51385 CUI9P3 66562388 EC50 = 64565.42 nM T51385 C7D0FE 66562389 EC50 = 8317.64 nM T51385 C1RBT5 66562390 EC50 = 5754.4 nM T51385 CD0GO5 66562391 EC50 > 100000 nM T51385 CI7WO1 66562392 EC50 = 3162.28 nM T51385 CAU1G2 66562488 EC50 = 1174.9 nM T51385 C6NIF3 67072752 EC50 = 776.25 nM T51385 C6RZL9 67134965 EC50 > 100000 nM T51385 C1PR6K 71655225 EC50 > 100000 nM T51385 CD6EU4 71655226 EC50 = 91201.08 nM T51385 C3XC7G 71655227 EC50 = 3890.45 nM T51385 CJMF15 71655293 EC50 = 3890.45 nM T51385 CD0AY7 73345869 EC50 = 1380.38 nM T51385 C75PUZ 73345870 EC50 = 300 nM T51385 CQ6N0O 73348895 EC50 = 300 nM T51385 CPF43O 73354950 EC50 = 300 nM T51385 CQ7T4B 73356514 EC50 = 300 nM T51385 CW1OF9 73776979 EC50 = 1000 nM T51385 CFG19U 73776995 EC50 = 440 nM T51385 C4P1AE 73776997 EC50 = 2100 nM T51385 CV78IM 73777065 EC50 = 3500 nM T51385 CPMI97 73777069 EC50 = 130 nM T51385 CC0V2Z 73777085 EC50 = 2100 nM T51385 CIX50H 73777111 EC50 = 1200 nM T51385 C9N7VS 73777135 EC50 = 360 nM T51385 CH5CY8 73777153 EC50 = 190 nM T51385 CAW6R9 73777156 EC50 = 200 nM T51385 C0PV3T 73777174 EC50 = 3100 nM T51385 CEYQ78 73777175 EC50 = 420 nM T51385 CI2DU6 82051616 EC50 = 972 nM T51385 CE36PD 82051652 EC50 = 251.19 nM T51385 C1PJ0B 84481843 EC50 = 1995.26 nM T51385 C54DHY 85470884 EC50 = 69 nM T51385 C5P9YL 85471695 EC50 = 142 nM T51385 C52UQK 85472222 EC50 = 1640 nM T51385 C6EZF9 85472225 EC50 = 25 nM T51385 COC7G3 85472227 EC50 = 31 nM T51385 C1ZV7R 85472359 EC50 = 34 nM T51385 CQ45DS 85472487 EC50 = 86 nM T51385 CFQ95A 85472618 EC50 = 71 nM T51385 CH03VU 85472621 EC50 = 104 nM T51385 COJ03Z 86280676 EC50 = 123.03 nM T51385 CPJ3C6 86281121 EC50 = 88 nM T51385 CJC2N4 86281122 EC50 = 40 nM T51385 C1AP9Y 86281123 EC50 = 50 nM T51385 C9UXT8 86281125 EC50 = 43 nM T51385 C6GWO5 86294762 EC50 = 179 nM T51385 CE5V2I 86343591 EC50 = 118 nM T51385 CU1S7W 86343594 EC50 = 156 nM T51385 C8MUH0 86343595 EC50 = 175 nM T51385 CW7J1F 86343790 EC50 = 923 nM T51385 C0FPW2 86343792 EC50 = 834 nM T51385 C30CKG 86343961 EC50 = 346 nM T51385 CI0CR7 86343963 EC50 = 448 nM T51385 CB85HZ 86343964 EC50 = 280 nM T51385 CWK6C4 86343965 EC50 = 134 nM T51385 CA24JF 86803193 EC50 > 10000 nM T51385 CNQ59Y 86803224 EC50 > 10000 nM T51385 CN9LT5 87054900 EC50 = 546 nM T51385 C3L9RY 87055315 EC50 = 200 nM T51385 C1CE7A 90404813 EC50 = 290 nM T51385 C86YLH 90405670 EC50 = 100 nM T51385 CPA9N8 90405989 EC50 = 145 nM T51385 C56QTC 90406219 EC50 = 161 nM T51385 C02IJY 90406228 EC50 = 117 nM T51385 CPC2Z8 90406335 EC50 = 262 nM T51385 CF80CZ 90406418 EC50 = 547 nM T51385 C34BXL 90406575 EC50 = 184 nM T51385 CHB6Z5 90406583 EC50 = 1370 nM T51385 C57DQV 90406631 EC50 = 112 nM T51385 CY74XR 90406842 EC50 = 164 nM T51385 CYH42M 90406893 EC50 = 877 nM T51385 CN91KF 90406961 EC50 = 162 nM T51385 CEN0W9 90406970 EC50 = 368 nM T51385 CN1RB5 90407027 EC50 = 533 nM T51385 C4S5AR 90407037 EC50 = 100 nM T51385 CJME80 90407263 EC50 = 91 nM T51385 CQ7RV3 90407441 EC50 = 173 nM T51385 CKD7O8 90407659 EC50 = 289 nM T51385 CSPL34 90417528 EC50 = 332 nM T51385 CPH7I9 90417978 EC50 = 51 nM T51385 C9H6RK 90418067 EC50 = 920 nM T51385 CC4YL3 90418139 EC50 = 132 nM T51385 CDJ1R8 90418278 EC50 = 42 nM T51385 CT95MO 90418333 EC50 = 75 nM T51385 CWVG94 90418476 EC50 = 51 nM T51385 CJ8XU6 90418513 EC50 = 56 nM T51385 CEH8J7 90418650 EC50 = 215 nM T51385 C7MJ4T 90418651 EC50 = 156 nM T51385 CQT1Z4 90418653 EC50 = 141 nM T51385 C0E8LZ 90418662 EC50 = 190 nM T51385 CU6L0Z 90418753 EC50 = 120 nM T51385 C25VYQ 90418782 EC50 = 173 nM T51385 CB7CG6 90418849 EC50 = 121 nM T51385 C2ZGD5 90418886 EC50 = 680 nM T51385 C04QKT 90442039 EC50 = 236 nM T51385 CQ58JG 90442468 EC50 = 197 nM T51385 CN17FZ 90644288 EC50 > 10000 nM T51385 CKH10I 91824000 EC50 = 12589.25 nM T51385 CZ6F7O 100493295 EC50 > 31622.78 nM T51385 CYVG83 100493305 EC50 > 31622.78 nM T51385 CYH40T 102338889 EC50 > 100000 nM T51385 CC1PY9 117734585 EC50 > 5000 nM T51385 CXPW86 117873187 EC50 = 2700 nM T51385 CR75CZ 117886639 EC50 = 3100 nM T51385 C6GAZ8 117886649 EC50 = 330 nM T51385 C53ZDS 118184919 EC50 = 332 nM T51385 CK09OQ 118707082 EC50 = 1000 nM T51385 CL0Q7T 118707083 EC50 = 501.19 nM T51385 CQV9Y5 118707084 EC50 = 398.11 nM T51385 CF98LS 118707085 EC50 > 31622.78 nM T51385 CQH32Z 118707086 EC50 > 31622.78 nM T51385 CC05JS 118707087 EC50 > 31622.78 nM T51385 CA72LW 118707088 EC50 > 31622.78 nM T51385 C4I7LM 118707170 EC50 > 31622.78 nM T51385 CS21LG 118707171 EC50 > 31622.78 nM T51385 C9XJ4H 118707172 EC50 > 31622.78 nM T51385 C4C8HP 118707173 EC50 = 316.23 nM T51385 CI28ZR 118707174 EC50 > 31622.78 nM T51385 CXKQ09 122184686 EC50 > 10000 nM T51385 CWDA29 127030344 EC50 = 33884.42 nM T51385 CZ6M9F 127030713 EC50 > 100000 nM T51385 CP60IR 127030714 EC50 > 100000 nM T51385 CQPG95 127030715 EC50 > 100000 nM T51385 C1P2AW 127031001 EC50 = 7585.78 nM T51385 CL24TF 127031002 EC50 = 34673.69 nM T51385 CMC5G3 127031003 EC50 = 17782.79 nM T51385 C32GDE 127031569 EC50 = 10471.29 nM T51385 CS9N8K 127033020 EC50 = 9549.93 nM T51385 CFZ6D3 127033352 EC50 = 4073.8 nM T51385 CG8LY9 127033353 EC50 = 4786.3 nM T51385 C2OM9J 127033354 EC50 > 100000 nM T51385 C6OPM1 127048827 EC50 > 10000 nM T51385 CH9S7P 127048842 EC50 > 10000 nM T51385 C6V3FP 127050770 EC50 > 10000 nM T51385 CE94RI 127051658 EC50 > 10000 nM T51385 C53BMN 134129938 EC50 = 11 nM T51385 C17CZB 134131620 EC50 = 55 nM T51385 CW4S6G 134131874 EC50 = 8.3 nM T51385 CO1RW6 134132142 EC50 = 94 nM T51385 CXE17Y 134132711 EC50 = 38.9 nM T51385 C4AB5J 134132951 EC50 = 43 nM T51385 CB89WY 134133275 EC50 = 102 nM T51385 C7DE1O 134133297 EC50 = 308 nM T51385 CG0L6Q 134133355 EC50 = 7.8 nM T51385 C2W0EY 134133675 EC50 = 290 nM T51385 C83GOA 134133797 EC50 = 1023.29 nM T51385 CS3P7G 134133992 EC50 = 79 nM T51385 CWS2G0 134134149 EC50 = 170 nM T51385 CJOQ95 134134229 EC50 = 16 nM T51385 CNA4L8 134134846 EC50 = 208.93 nM T51385 C96FRN 134135468 EC50 = 700 nM T51385 CCH39I 134136175 EC50 = 185 nM T51385 CPBG95 134136959 EC50 > 10000 nM T51385 C7VOB4 134137619 EC50 > 9950 nM T51385 CXRE49 134138099 EC50 = 436.52 nM T51385 CD9V6N 134138281 EC50 = 32 nM T51385 CN9LG1 134138318 EC50 = 498 nM T51385 C2J4UK 134138802 EC50 = 300 nM T51385 C5JM4L 134139171 EC50 = 68 nM T51385 CGO7M3 134140070 EC50 > 10000 nM T51385 C5SQU0 134140073 EC50 = 83 nM T51385 C76URI 134141029 EC50 = 97 nM T51385 CN9BG4 134141270 EC50 = 121 nM T51385 CJ30RW 134141489 EC50 > 10000 nM T51385 CI75ZW 134141650 EC50 = 5754.4 nM T51385 C6ZRV4 134142450 EC50 = 819 nM T51385 CCDO98 134142866 EC50 = 946 nM T51385 C4VL9A 134143163 EC50 = 182 nM T51385 CIN93P 134143370 EC50 = 170 nM T51385 CBLF04 134143899 EC50 = 544 nM T51385 C9QUR0 134144000 EC50 = 5 nM T51385 CBW12L 134144214 EC50 = 60 nM T51385 C0A8TH 134145071 EC50 = 16218.1 nM T51385 C2GH9K 134145195 EC50 > 9950 nM T51385 CYP7O1 134145412 EC50 = 66 nM T51385 C8C1DB 134145700 EC50 = 9 nM T51385 CU36BG 134145750 EC50 = 8174 nM T51385 C8KY5G 134145778 EC50 = 234.42 nM T51385 C96FUD 134146021 EC50 = 186 nM T51385 C9N5LO 134146386 EC50 = 42 nM T51385 CY3ZF0 134146590 EC50 > 10000 nM T51385 COYL20 134146720 EC50 = 13 nM T51385 CC13ZE 134146958 EC50 = 13 nM T51385 CO6N1L 134147107 EC50 = 2200 nM T51385 C1OMN0 134147174 EC50 = 188 nM T51385 CXH3T0 134147328 EC50 = 5248.07 nM T51385 CUO72N 134147601 EC50 = 130 nM T51385 CJ20TQ 134148110 EC50 = 21 nM T51385 C7XBW3 134148736 EC50 = 88 nM T51385 CQ5R4P 134149615 EC50 = 77 nM T51385 CA5B2J 134150245 EC50 = 57 nM T51385 C1GDK0 134150871 EC50 > 10000 nM T51385 CLM9Q7 134151115 EC50 = 153 nM T51385 CAG0Y1 134151150 EC50 > 10000 nM T51385 CRH0A7 134151903 EC50 = 130 nM T51385 CAY73T 134152336 EC50 = 330 nM T51385 C3SFX4 134152545 EC50 = 1659.59 nM T51385 CNK25T 134152845 EC50 > 9950 nM T51385 CRGW59 134153067 EC50 = 2691.53 nM T51385 CW54AS 134153222 EC50 = 1258.93 nM T51385 CVOE51 134153298 EC50 = 8 nM T51385 C7U9SB 134153546 EC50 = 230 nM T51385 C4H8UV 134153562 EC50 = 20 nM T51385 C4O0ZM 134153986 EC50 = 33 nM T51385 C49FKZ 134154330 EC50 = 2999 nM T51385 CV1E3G 134154415 EC50 = 5.6 nM T51385 C0GYX7 134154417 EC50 = 204 nM T51385 CM69QG 134154473 EC50 = 10 nM T51385 CZ98TW 134154643 EC50 > 10000 nM T51385 C6SA1G 134154953 EC50 = 2630.27 nM T51385 C69YFE 134154975 EC50 = 16595.87 nM T51385 CK29QG 134155067 EC50 = 6.2 nM T51385 C9LNQ5 134155277 EC50 = 254 nM T51385 CSM4R6 134155480 EC50 = 17 nM T51385 CA6RE0 134155847 EC50 = 17 nM T51385 C7TO6A 134155950 EC50 = 17 nM T51385 CK9M4A 134156096 EC50 = 198 nM T51385 CL92ZI 134156455 EC50 = 84 nM T51385 CA49BH 134156727 EC50 = 24 nM T51385 C7GDP1 134157207 EC50 = 149 nM T51385 CJ6T8B 134157563 EC50 = 474 nM T51385 C2GKN8 134157586 EC50 = 100 nM T51385 CJ1LT0 137631654 EC50 > 17000 nM T51385 CQS26D 137631865 EC50 = 350 nM T51385 CK8TZ6 137632299 EC50 = 110 nM T51385 C7TA3H 137632403 EC50 = 1992 nM T51385 CKD6O9 137632610 EC50 = 4800 nM T51385 C78BAZ 137633489 EC50 = 2000 nM T51385 C1GXR8 137633528 EC50 > 5000 nM T51385 C7MF0A 137633536 EC50 = 299 nM T51385 C68SZA 137634330 EC50 > 10000 nM T51385 C5DNV4 137634829 EC50 = 81 nM T51385 CGE59Q 137634844 EC50 = 9660 nM T51385 C1MPK7 137635671 EC50 = 71 nM T51385 CZ1OD2 137636167 EC50 = 722 nM T51385 CGH98J 137636217 EC50 = 1070 nM T51385 C3AI4N 137636575 EC50 = 71 nM T51385 CMO1E3 137636733 EC50 = 236 nM T51385 CL7BI1 137637243 EC50 = 990 nM T51385 CR53AY 137637576 EC50 = 60 nM T51385 C1MDE5 137637713 EC50 = 690 nM T51385 C5AR3F 137638176 EC50 = 410 nM T51385 CB0MZ3 137638317 EC50 = 720 nM T51385 C5UQ4L 137638318 EC50 = 740 nM T51385 CMPD78 137638355 EC50 = 188 nM T51385 CT93OE 137638911 EC50 = 630.96 nM T51385 CW7Y0B 137638939 EC50 > 17000 nM T51385 CGD21L 137638995 EC50 = 501.19 nM T51385 C5AXI9 137639797 EC50 > 5000 nM T51385 C29YVT 137640163 EC50 = 12000 nM T51385 C4JOD5 137640323 EC50 = 9977 nM T51385 CRZ2Y1 137640328 EC50 = 140 nM T51385 C68DOG 137640701 EC50 = 130 nM T51385 CE9Z4L 137641343 EC50 = 158.49 nM T51385 CDS7R1 137641818 EC50 = 250 nM T51385 CTW8I6 137642184 EC50 = 5911 nM T51385 CQC25W 137642248 EC50 = 4600 nM T51385 CZ4KW8 137642604 EC50 = 199.53 nM T51385 CNKP70 137642920 EC50 = 100 nM T51385 CABQ57 137643146 EC50 = 57 nM T51385 CM67CB 137643228 EC50 = 1130 nM T51385 CS59FT 137643339 EC50 = 362 nM T51385 CE59XO 137643731 EC50 = 470 nM T51385 C78MEF 137643958 EC50 = 120 nM T51385 CKD4H5 137645249 EC50 = 510 nM T51385 C2I9LX 137645347 EC50 = 220 nM T51385 CAOR76 137645556 EC50 > 17000 nM T51385 C4FM9C 137646094 EC50 > 5000 nM T51385 C2G5QA 137646145 EC50 = 1750 nM T51385 CM2C7J 137646188 EC50 = 2292 nM T51385 C4O8UV 137646368 EC50 = 2600 nM T51385 C7Y9PC 137646553 EC50 = 50.12 nM T51385 C4A0EY 137646995 EC50 = 150 nM T51385 CRTL26 137647294 EC50 = 2830 nM T51385 CQC17M 137647721 EC50 = 11380 nM T51385 CMQ47R 137647888 EC50 > 17000 nM T51385 CA5N8S 137648785 EC50 = 69 nM T51385 C8W7UQ 137648938 EC50 = 360 nM T51385 C61GUE 137649360 EC50 = 190 nM T51385 CD2E6Z 137649363 EC50 = 4100 nM T51385 CL1HE5 137649416 EC50 = 898 nM T51385 CV4T6F 137649555 EC50 = 640 nM T51385 C3JC2W 137649832 EC50 > 17000 nM T51385 C8KPQ5 137650498 EC50 = 2400 nM T51385 CMLH80 137651153 EC50 = 760 nM T51385 C6HT7R 137651358 EC50 = 600 nM T51385 C2OVI7 137651638 EC50 = 260 nM T51385 CLQ3W0 137652399 EC50 = 4300 nM T51385 C5BPA0 137653883 EC50 = 1450 nM T51385 CFI68P 137653903 EC50 > 10000 nM T51385 C47DPT 137653973 EC50 = 10000 nM T51385 C7P5OE 137654131 EC50 = 78 nM T51385 CO2L0W 137654721 EC50 = 251.19 nM T51385 C6B1NS 137655521 EC50 = 170 nM T51385 COB6K3 137656526 EC50 = 630.96 nM T51385 C3X5QA 137656733 EC50 = 900 nM T51385 CGA47X 137656909 EC50 > 17000 nM T51385 CN7I4Y 137657488 EC50 = 120 nM T51385 CQ50IA 137657736 EC50 = 1440 nM T51385 CIXP07 137657813 EC50 = 520 nM T51385 CKP08V 137657968 EC50 = 160 nM T51385 CK9R6S 137657972 EC50 = 39.81 nM T51385 CSR4W2 137658634 EC50 = 60 nM T51385 CXS6E7 137658977 EC50 = 470 nM T51385 CBG58K 137659266 EC50 > 10000 nM T51385 CAWH82 137659366 EC50 = 710 nM T51385 CP94BK 137659555 EC50 > 30000 nM T51385 CU9O2S 137660172 EC50 = 4000 nM T51385 CQU17B 137660302 EC50 = 400 nM T51385 CV56DT 137660451 EC50 = 150 nM T51385 CZR62H 137661388 EC50 = 304 nM T51385 C4AM0P 137661886 EC50 = 160 nM T51385 C45FZP 145955668 EC50 = 106 nM T51385 C2O3LF 145955958 EC50 > 10000 nM T51385 CR9J8V 145957609 EC50 > 10000 nM T51385 CZ8E7J 145959985 EC50 > 10000 nM T51385 CZC87F 145960576 EC50 = 99 nM T51385 CMJ50D 145961418 EC50 > 10000 nM T51385 CS9OA7 145965948 EC50 = 195.6 nM T51385 CB57ZL 145967268 EC50 = 396.2 nM T51385 CX4BD7 145967778 EC50 = 63.1 nM T51385 CD3K2O 145971522 EC50 = 94 nM T51385 CD67EV 145978633 EC50 = 126.8 nM T51385 CF34ZO 145982616 EC50 > 100000 nM T51385 CO8K0Z 145983493 EC50 = 186 nM T51385 CAEZ16 145983824 EC50 = 24040 nM T51385 CK9B5S 145984009 EC50 = 463 nM T51385 C0OJ2P 145984445 EC50 = 5039 nM T51385 CT9V1W 145984594 EC50 = 220 nM T51385 CKEB40 145984796 EC50 = 93 nM T51385 C0F2AH 145985122 EC50 = 638 nM T51385 C5C4YM 145985219 EC50 = 874 nM T51385 CIGK40 145985686 EC50 = 69 nM T51385 C5J4SE 145985748 EC50 = 347 nM T51385 CX9U0T 145986046 EC50 = 1478 nM T51385 C28DAN 145986262 EC50 = 2780 nM T51385 D01CCG 25150014 EC50 = 1445.44 nM T51385 D01VIX 73777063 EC50 = 66 nM T51385 D03JPL 79034 EC50 > 100000 nM T51385 D03LOG 5280450 EC50 = 316.23 nM T51385 D08MLH 46941175 EC50 = 6309.57 nM T51385 D08ZYC 11595431 EC50 = 1412.54 nM T51385 D0C5SV 5280934 EC50 = 2600 nM T51385 D0K6EG 57522038 EC50 = 43.65 nM T51385 D0N0UC 3893 EC50 = 7585.78 nM T51385 D0N9SV 25098573 EC50 = 1200 nM T51385 D0S0QY 66553168 EC50 = 933.25 nM T51385 D0T2CG 94216 EC50 > 100000 nM T51385 D0T4BP 97783 EC50 > 100000 nM T08231 C2IGS5 9831164 IC50 = 980 nM T08231 CD87QK 10121801 IC50 = 950 nM T08231 C9L2UX 10122216 IC50 = 2000 nM T08231 CSUI41 10168223 IC50 = 410 nM T08231 C4EUC3 10189472 IC50 = 2000 nM T08231 CEN82K 10211864 IC50 = 1300 nM T08231 C20FGH 10233020 IC50 = 1300 nM T08231 CM7H2R 10233142 IC50 = 1600 nM T08231 CER43X 10233451 IC50 = 1900 nM T08231 CPRC34 10233559 IC50 = 750 nM T08231 CZ7TP4 10233786 IC50 = 1300 nM T08231 C49OTB 10282988 IC50 = 1800 nM T08231 CS3DV6 10303703 IC50 = 810 nM T08231 CK80OJ 10304088 IC50 = 1100 nM T08231 C3NJ2U 10304660 IC50 = 1600 nM T08231 CS3Y6X 10304727 IC50 = 1800 nM T08231 CLQ0A4 10305142 IC50 = 2600 nM T08231 CP6VM4 22293649 IC50 = 1400 nM T08231 C5H1DR 22293657 IC50 = 900 nM T08231 CCV37T 22293696 IC50 = 1100 nM T08231 CBQN59 22293722 IC50 = 1500 nM T08231 C20MGL 22293806 IC50 = 930 nM T08231 CU3XR0 22293870 IC50 = 4400 nM T08231 CS9LH6 22293909 IC50 = 1400 nM T08231 CS1NY3 44410075 IC50 = 2700 nM T04413 D0E3TC 44259 IC50 = 4.32 nM T04413 D0T3ME 156422 IC50 > 30000 nM T04413 CACS26 11561968 Ki > 2000 nM T04413 CU0E8O 11690457 Ki > 2000 nM T04413 CLZ23U 24951610 IC50 = 8900 nM T04413 C2KY1G 25094210 IC50 > 10000 nM T04413 C6BWZ8 25145145 IC50 > 100 nM T04413 C78YWA 25145716 IC50 > 500 nM T04413 COTJ39 46863083 IC50 = 12000 nM T04413 CLS29B 46872626 IC50 > 10000 nM T04413 CXA03W 52920796 IC50 > 100 nM T04413 C6OTY5 53251320 IC50 > 30000 nM T04413 CE8OY2 53317913 IC50 > 100 nM T04413 C8NA4L 53384644 IC50 > 30000 nM T04413 C0UDY9 57401151 IC50 > 30000 nM T04413 C6BPR2 58985201 IC50 > 30000 nM T04413 C1MR8Q 60097495 IC50 > 1000 nM T04413 CV63UL 67240318 IC50 > 10000 nM T04413 CAU45T 91971978 IC50 > 30000 nM T04413 CDNC31 145967951 IC50 > 500 nM T04413 C2MD1Q 155513187 IC50 > 10000 nM T04413 D00ERW 44444843 Ki > 1526 nM T04413 D0E7VO 59627005 IC50 = 30.6 nM T04413 D0ME9B 46868971 IC50 > 10 nM T79570 D05VZE 119031 IC50 = 10000 nM T79570 D0G1LL 74221072 IC50 = 2 nM T79570 D0N6ZA 74221131 IC50 = 14 nM T79570 D0UM5R 74221070 IC50 = 7 nM T79570 D0T9HG 132519 IC50 = 480 nM T79570 CT8PU3 3671894 IC50 = 2400 nM T79570 C1FZ7Q 7257957 IC50 = 1100 nM T79570 CJS23I 9868333 Ki = 4600 nM T79570 C9X0YR 9954867 IC50 = 3 nM T79570 CN76XI 9957653 IC50 = 1000 nM T79570 CUA65C 9982414 IC50 = 8.1 nM T79570 CVK61T 10116047 IC50 = 1.4 nM T79570 CHUA34 10160545 IC50 > 1000 nM T79570 C4FSU0 10203714 IC50 = 330 nM T79570 C92BVJ 10223963 IC50 = 55 nM T79570 CV5X8A 10224181 IC50 > 25000 nM T79570 CU67RC 10275101 IC50 = 40 nM T79570 CY08WJ 10322755 Ki = 4600 nM T79570 CW1E7L 10667540 IC50 = 4300 nM T79570 CP17ID 11284983 IC50 = 5600 nM T79570 C8C5AV 11294179 Ki = 6700 nM T79570 CS8RH5 11295121 IC50 = 86 nM T79570 CLH50U 11318841 IC50 = 4400 nM T79570 C0XR3B 11330861 IC50 = 14300 nM T79570 COS67B 11456566 IC50 = 15000 nM T79570 C7QF0G 11467517 IC50 = 2200 nM T79570 CA2UB1 11487570 IC50 = 11600 nM T79570 C3RJ8Z 11496896 IC50 = 700 nM T79570 CWGN51 11510805 IC50 = 1100 nM T79570 C84OUY 11526630 IC50 = 900 nM T79570 C5MO0U 11526826 IC50 = 90 nM T79570 CD30LP 11532652 IC50 = 1200 nM T79570 CRF85U 11532881 IC50 = 1600 nM T79570 CB9SA2 11541301 IC50 = 590 nM T79570 CW5A4S 11569716 IC50 = 230 nM T79570 CVKA85 11570055 IC50 = 400 nM T79570 CB4MV2 11576629 IC50 = 1000 nM T79570 CW81GA 11598411 IC50 = 350 nM T79570 C0VCJ8 11613810 IC50 = 80 nM T79570 CYG73L 11635298 IC50 = 730 nM T79570 C1U9WL 11648679 IC50 = 430 nM T79570 CE4O0F 11676913 IC50 = 1700 nM T79570 C6T3SV 11678318 IC50 = 230 nM T79570 CV65NX 11685101 IC50 = 180 nM T79570 CRF7V9 11691964 IC50 = 100 nM T79570 C1K0LM 11720790 IC50 = 1900 nM T79570 C6HV8Z 11752434 IC50 = 1.1 nM T79570 CB80OT 12000718 IC50 = 2400 nM T79570 C43PJZ 12000720 IC50 = 7000 nM T79570 C6Y7QT 16664963 IC50 = 44000 nM T79570 C1F3NK 20725561 IC50 = 21 nM T79570 CIC4S9 22004232 IC50 = 3300 nM T79570 CXEP14 24754176 IC50 > 22000 nM T79570 CSQ9E4 24754248 IC50 > 22000 nM T79570 CX16GL 24754251 IC50 > 22000 nM T79570 COY8K0 24754252 IC50 = 10500 nM T79570 CZ7OA9 24901472 IC50 = 3000 nM T79570 CB4JP5 24901473 IC50 > 100000 nM T79570 CAB0Z9 24901474 IC50 = 30000 nM T79570 CYB16Q 24901475 IC50 = 50000 nM T79570 CNL70E 24901476 IC50 = 20000 nM T79570 CQD72G 24901477 IC50 = 9000 nM T79570 CQ51FL 24901478 IC50 = 4600 nM T79570 C4FI5C 24901479 IC50 > 100000 nM T79570 C1IO3Z 24901480 IC50 = 100000 nM T79570 C5SV4Y 24901482 IC50 = 2800 nM T79570 C3TW6N 24901483 IC50 = 1600 nM T79570 CE4C3B 24901484 IC50 = 12000 nM T79570 C6F0ZP 24901485 IC50 = 7500 nM T79570 CO4XQ7 24901486 IC50 = 1400 nM T79570 C27AKV 24901487 IC50 = 3800 nM T79570 C4Q3RF 24901488 IC50 = 400 nM T79570 CB94KU 24958549 IC50 > 22000 nM T79570 CU3W7Y 24960377 IC50 = 1900 nM T79570 CVR52U 25066764 IC50 > 5 nM T79570 CHR2P1 25183768 Ki > 25000 nM T79570 CCI64J 44224245 IC50 = 18000 nM T79570 CDG2K7 44393747 IC50 > 1000 nM T79570 CWUV21 44393760 IC50 > 1000 nM T79570 CQ6WZ5 44393836 IC50 > 1000 nM T79570 CR58XA 44393837 IC50 > 1000 nM T79570 CIH8T9 44393838 IC50 = 220 nM T79570 CK95WI 44393841 IC50 = 100 nM T79570 CAC72Q 44393867 IC50 = 100 nM T79570 CFR4G2 44393892 IC50 > 1000 nM T79570 CMBJ97 44393897 IC50 > 1000 nM T79570 CF3M5K 44393910 IC50 = 87 nM T79570 C4YJI9 44393913 IC50 = 26 nM T79570 C0E8BQ 44393936 IC50 = 370 nM T79570 CGU63Q 44393964 IC50 > 1000 nM T79570 C8P0IG 44393980 IC50 = 140 nM T79570 CP24NE 44394027 IC50 > 1000 nM T79570 CHP81Z 44394038 IC50 > 1000 nM T79570 CKB7S1 44394067 IC50 > 1000 nM T79570 CZB81D 44395506 IC50 = 1 nM T79570 CWGQ46 44404503 IC50 = 8600 nM T79570 CLXM58 44404504 IC50 > 15000 nM T79570 C30DKN 44404553 IC50 = 580 nM T79570 CIC60V 44406452 IC50 = 700 nM T79570 C4NK7V 44432463 IC50 = 7500 nM T79570 C47XUD 44571675 IC50 > 50000 nM T79570 CGF93P 44574388 IC50 = 800 nM T79570 C1U7CW 44574389 IC50 = 400 nM T79570 C9Z2DB 44574390 IC50 = 200 nM T79570 CFPS68 44574391 IC50 = 200 nM T79570 CE0CG7 44574578 IC50 = 3200 nM T79570 CA3F2R 44574579 IC50 = 20000 nM T79570 C5QY9R 44574666 IC50 = 5200 nM T79570 C1EGN9 44574994 IC50 = 700 nM T79570 CX7GV3 44575039 IC50 = 1800 nM T79570 CUJI69 44575089 IC50 = 4900 nM T79570 CBK40V 44575090 IC50 = 6000 nM T79570 CSX5I9 46175170 IC50 = 4 nM T79570 C9XQZ2 46845568 IC50 = 210 nM T79570 CE05DO 46848243 IC50 = 88 nM T79570 CI9JP2 46848247 IC50 = 158 nM T79570 CJ71XO 46848423 IC50 = 518 nM T79570 C8AO4U 46848424 IC50 = 1700 nM T79570 CKHU90 46848769 IC50 = 5500 nM T79570 CY8U6Z 46848942 IC50 = 8500 nM T79570 C39NMP 46848943 IC50 = 81 nM T79570 CZP4W7 46849587 IC50 = 60 nM T79570 CDV62X 46849588 IC50 = 163 nM T79570 CUX0Q1 46849589 IC50 = 284 nM T79570 C7IXV6 46849757 IC50 = 10 nM T79570 CDAJ65 46849758 IC50 = 60 nM T79570 C4H2IU 46849760 IC50 = 181 nM T79570 C5T3BD 46849926 IC50 = 61 nM T79570 CO5R2C 46849928 IC50 = 14 nM T79570 C7ECT5 46850266 IC50 = 3000 nM T79570 C97PJR 46850267 IC50 = 3000 nM T79570 CU54MG 46850268 IC50 > 10000 nM T79570 CTD23L 46850269 IC50 = 102 nM T79570 CQ1P2R 46850270 IC50 = 8 nM T79570 C59TML 46850431 IC50 = 6 nM T79570 C6SNA2 46850432 IC50 = 64 nM T79570 CT1WJ0 46850434 IC50 = 23 nM T79570 COD8N5 46850607 IC50 = 63 nM T79570 CV12IR 46850782 IC50 = 43 nM T79570 CTZA93 46850784 IC50 = 1817 nM T79570 C14PIN 49831179 IC50 > 30000 nM T79570 CUD7O0 50941549 IC50 = 23 nM T79570 CX8N4D 50990920 IC50 = 3.5 nM T79570 CXF4V3 50990921 IC50 = 0.69 nM T79570 C6U2CK 52945850 IC50 = 12000 nM T79570 C7CV6M 52947039 IC50 = 8000 nM T79570 C28MDL 52947079 IC50 > 30000 nM T79570 CMQZ70 53242178 IC50 = 26 nM T79570 C4L6ES 53317617 IC50 = 3.8 nM T79570 CB09MA 53318910 IC50 = 7.3 nM T79570 C47DIU 53318911 IC50 = 0.18 nM T79570 CC6DR2 53318912 IC50 = 0.48 nM T79570 C7V1NC 53320225 IC50 = 0.49 nM T79570 CVH2B7 53320226 IC50 = 4.2 nM T79570 CO8QK2 53320227 IC50 = 0.57 nM T79570 CNS3F2 53321542 IC50 = 0.52 nM T79570 C2O5KJ 53322874 IC50 = 1.1 nM T79570 C8KQY4 53322875 IC50 = 2200 nM T79570 C1N2BX 53322876 IC50 = 0.48 nM T79570 CSYW40 53322877 IC50 = 1.9 nM T79570 CGUC59 53322878 IC50 = 0.26 nM T79570 C3QHA6 53322879 IC50 = 0.68 nM T79570 C1VNZ9 53324198 IC50 = 1 nM T79570 C0H7FQ 53324260 IC50 = 5.4 nM T79570 CU7YG9 53325497 IC50 = 0.48 nM T79570 C4G1HK 53325498 IC50 = 0.94 nM T79570 CO5L1I 53325499 IC50 = 0.43 nM T79570 CZA03W 53326760 IC50 = 0.36 nM T79570 CM53CG 53326761 IC50 = 2.1 nM T79570 CWR6T4 53326860 IC50 = 2.8 nM T79570 CSUW40 54352406 IC50 = 2100 nM T79570 C3M8GZ 54580051 IC50 = 18 nM T79570 CL0WM9 54580052 IC50 = 11 nM T79570 CK26XF 54580053 IC50 = 51 nM T79570 CA6K5D 54581029 IC50 = 1.9 nM T79570 C8PE1G 54581030 IC50 = 530 nM T79570 CVK72M 54582073 IC50 = 4.5 nM T79570 CBK18O 54582074 IC50 = 48 nM T79570 CP2F1B 54582075 IC50 = 9.7 nM T79570 CZNU23 54582076 IC50 = 19 nM T79570 C0U5HZ 54582077 IC50 = 20 nM T79570 CSTG96 54582078 IC50 = 92 nM T79570 C8SG9Y 54582079 IC50 = 1.4 nM T79570 CZI6S3 54582080 IC50 = 110 nM T79570 CY50KX 54582081 IC50 = 1.2 nM T79570 CH6Q2Z 54583016 IC50 = 16 nM T79570 C3V9LQ 54583017 IC50 = 470 nM T79570 CT80KQ 54583018 IC50 = 5.6 nM T79570 CPT4L5 54583019 IC50 = 380 nM T79570 CBEV27 54584024 IC50 = 5.8 nM T79570 CM87DP 54584025 IC50 = 100 nM T79570 C3JY9Z 54584969 IC50 = 4.1 nM T79570 CBJ5U9 54584970 IC50 = 8.7 nM T79570 CI5W2A 54585926 IC50 = 91 nM T79570 C28GKQ 54585927 IC50 = 13 nM T79570 CAZ76E 54586892 IC50 = 29 nM T79570 CM0OQ3 54586893 IC50 = 10 nM T79570 CK1NS7 54586894 IC50 = 20 nM T79570 CMC4Y1 54586895 IC50 = 24 nM T79570 C2MKX5 54586896 IC50 = 400 nM T79570 CU91QP 54586897 IC50 = 52 nM T79570 CI08RQ 54586898 IC50 = 2.7 nM T79570 C6PRI4 54586899 IC50 = 130 nM T79570 C9UJ8H 54586903 IC50 = 210 nM T79570 CKR9V8 56659819 IC50 = 3300 nM T79570 CL0U6N 56663282 IC50 = 9700 nM T79570 CI80OC 56670131 IC50 = 1200 nM T79570 CO2NY6 56670132 IC50 = 4900 nM T79570 CK47BT 56928417 IC50 = 310 nM T79570 C9GA0X 57390229 IC50 = 2100 nM T79570 C0IU4S 57390230 IC50 = 500 nM T79570 C8MSI6 57390231 IC50 = 30000 nM T79570 CLI26N 57390232 IC50 = 33000 nM T79570 CCN3K2 57390233 IC50 = 4700 nM T79570 CJ49DO 57390234 IC50 = 9100 nM T79570 CU34JA 57390237 IC50 = 3700 nM T79570 C9SD5O 57390259 IC50 = 540 nM T79570 C40GSM 57392019 IC50 = 8400 nM T79570 C6N3QB 57392020 IC50 > 200000 nM T79570 C0UXZ5 57392021 IC50 = 25000 nM T79570 CJC7M9 57392022 IC50 = 8500 nM T79570 CAL94F 57392025 IC50 = 760 nM T79570 CA6L5W 57392045 IC50 = 1900 nM T79570 CEGL19 57393743 IC50 > 200000 nM T79570 CB64TD 57393744 IC50 = 5500 nM T79570 CV3W5X 57393745 IC50 = 10600 nM T79570 C3CA9G 57393746 IC50 = 1400 nM T79570 CZBL73 57395457 IC50 = 7200 nM T79570 C27AQN 57395458 IC50 = 800 nM T79570 C10PRG 57395459 IC50 = 2400 nM T79570 C42XNM 57395460 IC50 = 15000 nM T79570 C17DMO 57395461 IC50 = 800 nM T79570 CZX7S9 57395466 IC50 = 22000 nM T79570 CQ4JU6 57395492 IC50 = 2700 nM T79570 CXI12G 57397306 IC50 = 40000 nM T79570 CVP2M7 57397307 IC50 = 50000 nM T79570 CR6GS0 57397308 IC50 > 75000 nM T79570 CBY21D 57397314 IC50 = 400 nM T79570 C43OUK 57398988 IC50 = 20000 nM T79570 C5R4TH 57398989 IC50 = 15000 nM T79570 C9CH0P 57398990 IC50 = 4100 nM T79570 CR59KW 57398991 IC50 = 420 nM T79570 C27HQG 57400706 IC50 = 100000 nM T79570 C08PQO 57400707 IC50 = 5600 nM T79570 C5U9NO 57400708 IC50 = 2200 nM T79570 C3T2CY 57402479 IC50 = 100000 nM T79570 CFCZ78 57402480 IC50 = 13200 nM T79570 CR94TK 57402481 IC50 = 8200 nM T79570 COP3C5 57402482 IC50 = 1400 nM T79570 C6HZ1P 57402483 IC50 = 1000 nM T79570 CGMQ47 57402485 IC50 = 2600 nM T79570 C37JZN 57402486 IC50 = 420 nM T79570 C52ESR 66559934 IC50 = 1870 nM T79570 C57ARI 66560021 IC50 = 1500 nM T79570 CU58DB 66560022 IC50 = 6000 nM T79570 C16RDM 66560389 IC50 = 8300 nM T79570 C8RZG9 66560479 IC50 = 1200 nM T79570 CHGS62 70218785 IC50 = 333 nM T79570 C5W2UN 70218786 IC50 = 370 nM T79570 CSMG89 70220118 IC50 = 30 nM T79570 C16KXI 70221056 IC50 = 5600 nM T79570 C4WA8U 70222009 IC50 > 10000 nM T79570 CKW2Q5 71453375 IC50 = 1300 nM T79570 CNX9B1 71652215 IC50 = 630 nM T79570 C7RZN9 71652216 IC50 = 3500 nM T79570 C0NTU7 71652382 IC50 = 5800 nM T79570 CA5XS1 71652383 IC50 = 80 nM T79570 CGQK53 73346500 IC50 = 1400 nM T79570 CMO17L 73346503 IC50 = 1000 nM T79570 CW01EA 73349535 IC50 = 630 nM T79570 CE79UD 73349536 IC50 = 2900 nM T79570 CI63PO 73351092 IC50 = 730 nM T79570 C82OGI 73352555 IC50 = 1500 nM T79570 CK8U6F 73352557 IC50 = 2000 nM T79570 CBZE87 73354044 IC50 = 610 nM T79570 C75IRY 73354046 IC50 = 1600 nM T79570 C8WC1K 73355580 IC50 = 790 nM T79570 CA5T7P 73603957 IC50 = 2 nM T79570 C8VN1R 74221194 IC50 = 1 nM T79570 CUE7G4 86287514 IC50 = 74 nM T79570 CGQ8F3 86287515 IC50 = 8 nM T79570 CJ37XE 86287516 IC50 = 3 nM T79570 CO2FL5 90137145 IC50 = 4 nM T79570 CRT54C 101910871 IC50 = 4 nM T79570 C6VD3T 118722685 IC50 = 110 nM T79570 C5ZS4E 118722686 IC50 = 12 nM T79570 CIZB24 118722687 IC50 = 17 nM T79570 C5C0ZX 118722688 IC50 = 22 nM T79570 C7A9FK 122191851 IC50 = 6500 nM T79570 CTN42D 132941363 IC50 = 4 nM T79570 CWS84X 135937145 IC50 = 22 nM T79570 CJG54U 136219136 IC50 > 10000 nM T79570 C3CAV5 136219141 IC50 = 23000 nM T79570 CPB07Z 136241630 IC50 = 21000 nM T79570 CS80YI 137652598 IC50 = 12 nM T79570 CZ8H6N 137661550 IC50 = 6 nM T79570 CZ25LW 155512044 IC50 = 4 nM T79570 CP9YX2 155567218 IC50 = 6 nM T79570 C8D5VK 155567855 IC50 = 8 nM T79570 D0FD9M 54585928 IC50 = 1.2 nM T79570 D0H6CK 10160968 Ki = 1834 nM T79570 D0Y1NM 24901481 IC50 = 5500 nM T79501 CQEF34 1002773 IC50 > 100000 nM T79501 CIZF42 122178085 IC50 = 6000 nM T79501 C6KV9H 124081151 IC50 > 100000 nM T79501 CF29KH 134159782 IC50 = 20000 nM T79501 C4LK1X 137635057 IC50 > 50000 nM T79501 CDPN65 137661881 IC50 > 50000 nM T79501 CE58DF 153041236 IC50 > 100000 nM T79501 C7C8HI 155529624 IC50 > 30000 nM T79501 D09CLP 439155 IC50 > 50000 nM T79501 D09ENZ 56962336 IC50 = 7500 nM T07806 D01AZG 5073 Ki = 10 nM T07806 D01TSI 8223 Ki = 2.1 nM T07806 D03RZV 5504 Ki > 10000 nM T07806 D03WEX 9966051 Ki = 33 nM T07806 D04JEE 4946 EC50 > 5011.87 nM T07806 D06FPQ 77992 Ki = 10.3 nM T07806 D08VRO 3822 IC50 = 6500 nM T07806 D09EBS 4636 Ki = 0.3 nM T07806 D0F2PO 4828 Ki = 2600 nM T07806 D0G8NN 119570 Ki = 3508 nM T07806 D0H3HM 60795 Ki = 1000 nM T07806 D0H7KF 5002 Ki > 1000 nM T07806 D0NG7O 60857 Ki = 4.2 nM T07806 D0S9MU 5078 Ki = 10.1 nM T07806 D0T3KI 4440 Ki = 3.3 nM T07806 D0V4QS 135398745 Ki = 1000 nM T07806 D0WV3U 4893 Ki > 7700 nM T07806 D0Y4DY 5709 Ki = 13 nM T07806 D0Z1RV 135398737 Ki = 1000 nM T07806 D0Z6UC 5358 Ki = 5.5 nM T07806 D08CJK 1150 Ki = 36 nM T07806 D09GHO 5311258 Ki = 83 nM T07806 D0N1HW 5311200 Ki > 10000 nM T07806 D00OWF 5280953 Ki > 10000 nM T07806 D00NLD 9881526 IC50 = 1.3 nM T07806 D01WJZ 60820 Ki = 2880 nM T07806 D02ZSO 6426760 EC50 = 430 nM T07806 D06DZI 107780 Ki = 0.14 nM T07806 D07BCO 5684 Ki = 24 nM T07806 D07BUO 25067561 Ki = 12 nM T07806 D08XWZ 9860595 Ki = 610 nM T07806 D0B7SP 11292933 Ki = 3.162 nM T07806 D0K4PN 9830790 Ki = 1.7 nM T07806 D0OS6O 60149 Ki = 56 nM T07806 D0Q2JS 10436045 Ki = 12.59 nM T07806 D0QF4Z 196968 Ki = 0.3162 nM T07806 D0SU1F 132552 IC50 = 14.45 nM T07806 D0YP7L 6604889 Ki = 1000 nM T07806 C32BCH 4656 Ki = 1980 nM T07806 C5H9CN 9287 Ki = 501.19 nM T07806 CVD75F 20810 Ki = 7.4 nM T07806 CNZD18 36381 Ki > 10000 nM T07806 C0OZ3N 37732 Ki = 5960 nM T07806 CU1TN8 47570 Ki > 10000 nM T07806 CW2T4Y 78576 Ki > 30000 nM T07806 CB6G3Z 91536 Ki = 4100 nM T07806 CW9EY7 127036 Ki = 10 nM T07806 CFSE35 129503 Ki = 270 nM T07806 CD89VU 137235 Ki > 30000 nM T07806 CGT8R0 160510 Ki > 10000 nM T07806 CZ3N4E 178081 Ki = 364 nM T07806 COPZ85 188006 Ki = 7.8 nM T07806 COZK91 210076 Ki > 10000 nM T07806 CQ97BV 225047 Ki > 10000 nM T07806 CYV1R3 417052 Ki > 10000 nM T07806 C6NE2K 547517 Ki > 10000 nM T07806 CZN6S9 743974 EC50 > 31622.78 nM T07806 C2VLP8 752521 Ki = 1531 nM T07806 C7Y3LQ 1328538 Ki = 260 nM T07806 C5DU2K 2199302 Ki = 26 nM T07806 C7PM8O 2261792 Ki = 107 nM T07806 CNMB94 2574642 Ki > 10000 nM T07806 CB3M6V 2762737 Ki = 14.2 nM T07806 C3M7GN 3016908 Ki = 3480 nM T07806 C8R1IU 3604129 Ki = 94 nM T07806 CS8KE2 3649661 Ki > 10000 nM T07806 CW34VC 6160690 Ki = 0.2 nM T07806 C9EO4Z 6422277 Ki = 1225 nM T07806 CZV19U 6426761 IC50 = 83 nM T07806 C0QCK1 6918455 Ki = 794.33 nM T07806 CW0ZE5 6918542 Ki = 2200 nM T07806 CC5PQ0 6918601 Ki = 3100 nM T07806 C1WXY3 6918603 Ki = 1995.26 nM T07806 CD0Z4I 6918648 Ki = 794.33 nM T07806 CCT52F 9795333 Ki = 1570 nM T07806 CUD06Z 9796627 Ki = 420 nM T07806 CX7I8J 9802187 Ki = 203 nM T07806 CCV0M4 9802530 Ki = 28 nM T07806 CZL0O6 9803620 EC50 = 103000 nM T07806 CE0DI5 9804612 Ki = 316.23 nM T07806 C8XGV3 9804849 IC50 = 800 nM T07806 CNX4F0 9805456 Ki = 2511.89 nM T07806 CGJB47 9816035 Ki = 712 nM T07806 CH7U3C 9816604 Ki > 5000 nM T07806 CWOS30 9817810 Ki = 6.5 nM T07806 CPXI10 9826761 Ki = 67 nM T07806 C0AU9L 9826801 Ki = 48 nM T07806 CLU54H 9827354 Ki = 208 nM T07806 CWS18C 9832057 EC50 = 0.58 nM T07806 C3K4XT 9837108 Ki = 2780 nM T07806 CRW5N0 9837525 Ki = 37 nM T07806 C28HXY 9844873 IC50 = 15 nM T07806 CNB65K 9848303 Ki = 36 nM T07806 CDOG70 9848876 Ki = 28 nM T07806 CM13ZV 9856041 Ki > 10000 nM T07806 CNCK78 9862256 Ki = 11 nM T07806 C8ROC3 9866484 IC50 = 282 nM T07806 CB1F0C 9867475 Ki = 190 nM T07806 C57YPX 9867902 IC50 = 62 nM T07806 C3GMU5 9868889 Ki = 0.3 nM T07806 C7AB8O 9870053 Ki = 3162.28 nM T07806 C19VUG 9871977 Ki = 5.012 nM T07806 CK76MQ 9872238 Ki = 1.4 nM T07806 C35LIA 9881324 IC50 = 830 nM T07806 C1WF3D 9881478 Ki = 342 nM T07806 CZ6NK9 9881603 Ki = 4435 nM T07806 CJW1P5 9888494 Ki < 3981.07 nM T07806 C6N8UE 9889681 Ki = 316.23 nM T07806 CM52WU 9890119 Ki = 630.96 nM T07806 CF5GN4 9890331 IC50 = 56 nM T07806 CEG1K5 9891002 Ki = 501.19 nM T07806 C7QMK5 9891617 Ki = 1258.93 nM T07806 CEL29O 9891618 Ki = 501.19 nM T07806 C3J8GU 9892409 Ki = 3981.07 nM T07806 CFM67S 9897637 EC50 = 0.1 nM T07806 CUN81Q 9905249 Ki > 10000 nM T07806 CYWQ50 9906447 Ki > 10000 nM T07806 CYZ5N4 9909089 Ki = 0.1995 nM T07806 C3BR6W 9910451 Ki = 340 nM T07806 C4L2CV 9911120 IC50 = 3801.89 nM T07806 C9B3EA 9911844 Ki < 1000 nM T07806 C78MDV 9913554 Ki = 630.96 nM T07806 C4UYZ7 9927441 Ki = 2300 nM T07806 CJ6CF2 9928474 Ki = 2.3 nM T07806 CJS2T1 9930155 IC50 = 145 nM T07806 C5V0UE 9933975 Ki = 0.5 nM T07806 CYVZ47 9934284 Ki = 1000 nM T07806 CWO45F 9935387 Ki = 630.96 nM T07806 CYH3R7 9947817 Ki = 720 nM T07806 C41HSL 9948210 Ki = 939 nM T07806 CM5A2D 9949172 IC50 = 309 nM T07806 CN7A4C 9949568 Ki = 1862 nM T07806 C63EWV 9950390 Ki = 2300 nM T07806 CO49NV 9952249 IC50 = 0.5 nM T07806 CK8NR2 9954121 Ki = 1584.89 nM T07806 C48OKD 9954663 Ki = 440 nM T07806 C9QPM4 9955522 Ki = 0.631 nM T07806 CSK1B2 9955819 Ki = 0.3 nM T07806 CFR41N 9957068 Ki = 5011.87 nM T07806 CZ9SC7 9957274 Ki = 1 nM T07806 CGO64P 9957376 Ki = 5.012 nM T07806 CTZ4U0 9972838 Ki = 587 nM T07806 C2XG1I 9977716 Ki = 0.3981 nM T07806 CFN50J 9978683 Ki > 5000 nM T07806 CPX92V 9979309 Ki = 0.5012 nM T07806 CXZM08 9981270 Ki = 115 nM T07806 CCR0T4 9984109 EC50 = 0.28 nM T07806 CN3D8M 9994674 Ki = 38 nM T07806 C1RNF9 9995233 Ki = 303 nM T07806 CXI19F 9997421 Ki = 552 nM T07806 CSGQ91 9997422 Ki = 856 nM T07806 C8A6EZ 10001971 Ki = 0.631 nM T07806 CCE86A 10003971 Ki = 119 nM T07806 CV4T9U 10008868 Ki = 0.14 nM T07806 C4F5JB 10015980 Ki = 109 nM T07806 CV7IP3 10016747 Ki = 133 nM T07806 C8JFH0 10016864 Ki = 194 nM T07806 CV7R9F 10020040 Ki > 10000 nM T07806 CK18LT 10020895 Ki = 1200 nM T07806 C04ZAS 10021450 Ki = 56 nM T07806 CQHW51 10023176 Ki = 0.7943 nM T07806 CM7W9G 10024936 Ki = 50.12 nM T07806 CA7MG0 10044965 Ki = 11 nM T07806 C25WVJ 10047566 IC50 > 1000 nM T07806 C2UI7F 10048252 Ki = 150 nM T07806 CF84QJ 10048342 Ki = 0.7943 nM T07806 C8JLO2 10048343 Ki = 6.31 nM T07806 C5PQ2I 10060289 Ki = 20 nM T07806 C9ENY6 10062659 Ki = 142 nM T07806 CHQ1L3 10064361 Ki = 179 nM T07806 C0GI7T 10064500 Ki = 4605 nM T07806 C98DKQ 10065239 Ki = 618 nM T07806 C6DC9G 10065919 Ki = 1096 nM T07806 C2EG0W 10068933 Ki = 15.4 nM T07806 CXW80P 10069802 Ki = 11 nM T07806 CJM76I 10070281 Ki = 153 nM T07806 C9KWT3 10071738 Ki = 0.5012 nM T07806 CV6R2F 10073139 Ki = 0.3162 nM T07806 CVE2T1 10076176 IC50 = 100 nM T07806 CQ1YA4 10076876 Ki = 6.4 nM T07806 CIO9D1 10088038 Ki = 177 nM T07806 CR3D5E 10091430 IC50 = 6918.31 nM T07806 CIZ50V 10096890 Ki = 23 nM T07806 CB4W8T 10105889 IC50 = 5800 nM T07806 C2ISY6 10114480 Ki = 6.31 nM T07806 C9PG3D 10115847 Ki = 158.49 nM T07806 CJZX05 10115848 Ki = 1258.93 nM T07806 CP1CL5 10127149 Ki = 39.81 nM T07806 CLFA47 10127209 Ki = 1995.26 nM T07806 CKYQ52 10127424 Ki = 1.995 nM T07806 CRJ8M9 10127673 Ki = 6.31 nM T07806 C4SN0A 10127877 Ki = 7.943 nM T07806 C9J6KH 10128059 Ki = 39.81 nM T07806 CNA8W3 10130620 Ki = 6830 nM T07806 CXCY91 10131024 Ki = 47 nM T07806 CWMT35 10138727 Ki < 1000 nM T07806 C4X9RB 10150658 Ki = 251.19 nM T07806 CKGC73 10150796 Ki = 63.1 nM T07806 CJI9T7 10151492 Ki = 25.12 nM T07806 CSPG27 10159927 Ki = 100 nM T07806 C9JLX2 10161027 Ki = 794.33 nM T07806 CVA6N0 10161028 Ki = 19.95 nM T07806 C5DSA0 10163458 Ki = 1300 nM T07806 C2N0XG 10164215 Ki = 51 nM T07806 C5E4SQ 10172853 Ki = 158.49 nM T07806 C3YT8A 10173169 Ki = 251.19 nM T07806 CJRV76 10173263 Ki = 19.95 nM T07806 CMP89S 10173443 Ki = 39.81 nM T07806 CT0CX5 10174078 Ki = 3.981 nM T07806 CQXI36 10174088 Ki = 158.49 nM T07806 C34ROH 10174199 Ki = 1.259 nM T07806 CEDP29 10183895 Ki = 39.81 nM T07806 C6NA5G 10194297 Ki = 158.49 nM T07806 CI76JU 10194809 Ki = 15.85 nM T07806 CLHY30 10194820 Ki = 50.12 nM T07806 CW1CM3 10195275 Ki = 6.31 nM T07806 CNT0Y6 10198320 Ki = 600 nM T07806 CMWD23 10198756 Ki = 110 nM T07806 CE3S6M 10216160 Ki = 398.11 nM T07806 CRW49L 10216744 Ki = 63.1 nM T07806 C80QXD 10216873 Ki = 19.95 nM T07806 CQ7ND4 10220230 Ki = 800 nM T07806 CF4N1M 10237964 Ki = 19.95 nM T07806 C0Q2ZD 10238160 Ki = 630.96 nM T07806 CIR98N 10238565 Ki = 15.85 nM T07806 CK39BA 10238566 Ki = 1.995 nM T07806 C3L0WD 10238762 Ki = 63.1 nM T07806 CI9KH6 10238763 Ki = 125.89 nM T07806 CC36JL 10245352 Ki = 228 nM T07806 CK9NT0 10247448 Ki = 409 nM T07806 C4Q2SH 10249573 Ki = 3981.07 nM T07806 CD83JK 10251722 Ki = 2.3 nM T07806 CUSP67 10252256 IC50 = 49 nM T07806 CMRA02 10257042 Ki = 1000 nM T07806 CG5M3Z 10263828 Ki = 7660 nM T07806 C7DJ2O 10266598 Ki = 714 nM T07806 CH31DX 10267394 Ki > 10000 nM T07806 CTE91S 10267412 Ki = 196 nM T07806 CVC87R 10275633 Ki = 0.7943 nM T07806 CQ8N3F 10288132 Ki = 7.943 nM T07806 CT12FP 10299410 Ki = 30 nM T07806 C8XKC0 10310103 Ki = 200 nM T07806 C3G8KJ 10310285 Ki = 12.59 nM T07806 C0WRV9 10310423 Ki = 125.89 nM T07806 CU89JD 10314060 Ki > 10000 nM T07806 C0OJ2C 10319235 Ki = 0.631 nM T07806 CPH30X 10319737 Ki = 1.995 nM T07806 CXG6B1 10341129 Ki = 0.631 nM T07806 C4IA8Z 10341917 IC50 = 62 nM T07806 C0UTS5 10342552 Ki = 3 nM T07806 C9IAV3 10346043 Ki > 5011.87 nM T07806 CG0X4W 10356544 Ki = 789 nM T07806 C2J3OP 10358224 Ki = 121 nM T07806 CR53YS 10365683 Ki = 3.3 nM T07806 CM97GO 10370874 Ki = 3.162 nM T07806 C1P9DA 10376496 Ki = 483 nM T07806 CW7MQ0 10376578 Ki = 1.9 nM T07806 CPU8B2 10379784 Ki = 304 nM T07806 C61HZF 10379833 Ki = 49 nM T07806 C36TNW 10383010 Ki = 992 nM T07806 CMZA83 10383646 Ki > 5000 nM T07806 C0XG9M 10387420 Ki = 1.585 nM T07806 C1U7LS 10398118 Ki = 1512 nM T07806 C20KTU 10400189 Ki = 227 nM T07806 C3ESO4 10401862 Ki = 948 nM T07806 CQ5V6K 10402263 Ki = 26 nM T07806 CG60RT 10403260 Ki = 439 nM T07806 C9RZ1N 10403999 Ki = 70 nM T07806 CLEU45 10406614 Ki = 46 nM T07806 C8S3XE 10409556 IC50 = 3019.95 nM T07806 C4TPN1 10413595 Ki = 1258.93 nM T07806 CK1WH6 10424220 Ki = 216 nM T07806 CQ2Y4A 10425027 Ki = 1654 nM T07806 CR4LS0 10430623 Ki > 5000 nM T07806 CN58XF 10432512 Ki = 187 nM T07806 CD7U5I 10433930 Ki > 10000 nM T07806 CDU91R 10434550 Ki = 0.5 nM T07806 CBAY90 10445946 Ki = 270 nM T07806 C9S5WP 10449461 Ki = 249 nM T07806 C9WA5Q 10452875 Ki = 31.62 nM T07806 CFK16Y 10454806 Ki = 0.3981 nM T07806 CYMS64 10454807 Ki = 1 nM T07806 C57RFG 10456869 IC50 = 96 nM T07806 CYS76Z 10468376 Ki = 2275 nM T07806 C73TEG 10475893 Ki = 243 nM T07806 CL63TF 10477223 Ki = 2.512 nM T07806 CE9R8Z 10477461 IC50 = 30 nM T07806 CWY2J3 10478217 Ki = 0.5012 nM T07806 CEF2O6 10478367 Ki = 2 nM T07806 CPB1I5 10488933 Ki > 10000 nM T07806 C1XT2J 10490160 Ki > 10000 nM T07806 CVJ4I3 10494885 IC50 = 97.72 nM T07806 C0I3BG 10496545 Ki = 172 nM T07806 CQ9A2N 10498633 Ki = 135 nM T07806 C65KTM 10500370 IC50 = 87 nM T07806 C4IXZ5 10500422 Ki = 6.1 nM T07806 C9SV3J 10501944 IC50 = 32 nM T07806 C97AGV 10501945 IC50 = 74 nM T07806 C74XEH 10502669 IC50 = 39 nM T07806 CNGM74 10502763 IC50 = 165 nM T07806 C1ALS8 10502988 IC50 = 35 nM T07806 CD3IL2 10503687 EC50 = 440 nM T07806 CD47NC 10503731 IC50 = 47 nM T07806 CCM78N 10504095 IC50 = 200 nM T07806 CS1RN9 10504096 IC50 = 71 nM T07806 CY7OA9 10504097 IC50 = 98 nM T07806 CNUR81 10504600 IC50 = 13 nM T07806 C2FDP8 10505438 IC50 = 46 nM T07806 CFJ45P 10505525 IC50 = 8.9 nM T07806 CUT89L 10517352 Ki = 188 nM T07806 CCPO93 10518850 Ki = 14 nM T07806 CNAZ85 10519108 IC50 = 93 nM T07806 CCQA42 10525100 IC50 = 62 nM T07806 CT28NZ 10526567 IC50 = 95 nM T07806 CP16JO 10526642 IC50 = 270 nM T07806 CUWV98 10526736 IC50 = 98 nM T07806 CF47AX 10526737 IC50 = 930 nM T07806 CA15PT 10527882 IC50 = 48 nM T07806 CZLC18 10528410 IC50 = 6.2 nM T07806 C0ZM5P 10531639 Ki = 0.22 nM T07806 C5HEN4 10536129 Ki > 10000 nM T07806 C1F9QW 10537557 Ki > 10000 nM T07806 CI36TG 10539089 IC50 = 44.67 nM T07806 CE3OX5 10541847 Ki = 3865 nM T07806 CMIV90 10544144 Ki > 1000 nM T07806 CF8NY5 10546537 IC50 = 263.03 nM T07806 CN3EP8 10548444 IC50 = 36 nM T07806 CIKZ61 10549785 IC50 = 140 nM T07806 C8AC6N 10550488 IC50 = 420 nM T07806 CNR5F7 10550857 IC50 = 3.1 nM T07806 CYB74T 10551206 IC50 = 14 nM T07806 CXA12U 10551207 IC50 = 170 nM T07806 C4MP8V 10551328 EC50 = 510 nM T07806 C3UK0W 10551525 IC50 = 520 nM T07806 C8CGV9 10551857 IC50 = 210 nM T07806 CL9O3W 10552243 IC50 = 410 nM T07806 CUE54L 10552573 IC50 = 460 nM T07806 CX0N3A 10552663 IC50 = 10 nM T07806 CCVQ57 10560632 Ki = 66 nM T07806 CHOZ29 10567450 Ki = 35 nM T07806 CP53ZW 10571716 IC50 = 320 nM T07806 CJ2YD5 10572483 IC50 = 20 nM T07806 CP7AX5 10573843 IC50 = 13 nM T07806 CHE80N 10573876 Ki = 1000 nM T07806 C4Y1WU 10573904 IC50 = 3.3 nM T07806 CVI9U2 10574570 IC50 = 45 nM T07806 CMX1B0 10574671 IC50 = 18 nM T07806 CIB5V0 10574762 IC50 = 120 nM T07806 C5CR0T 10575553 EC50 = 810 nM T07806 CJC3R5 10575878 IC50 = 210 nM T07806 CWPE61 10576874 IC50 = 100 nM T07806 C09ZXH 10577268 Ki = 1.585 nM T07806 CA8NT1 10577311 IC50 = 24 nM T07806 CCG7A9 10584924 Ki = 1120 nM T07806 C5BV8A 10585509 Ki = 200 nM T07806 CWM6U4 10588458 Ki = 1205 nM T07806 C1O3LZ 10588665 IC50 = 9.55 nM T07806 CCBU34 10590370 Ki = 275 nM T07806 C0N2EP 10592083 IC50 = 63 nM T07806 CY3BD0 10592324 IC50 = 141.25 nM T07806 CJV2Z4 10596387 IC50 = 275 nM T07806 CITF30 10596566 IC50 = 27 nM T07806 CO23YX 10597140 Ki < 3162.28 nM T07806 C6I3LK 10597210 Ki = 12.59 nM T07806 C4Y2OD 10597901 IC50 = 120 nM T07806 CE3W5U 10597902 IC50 = 15 nM T07806 CW25KM 10600063 IC50 = 69 nM T07806 CKJZ76 10600212 IC50 = 380 nM T07806 C98XYU 10600213 IC50 = 310 nM T07806 CJ3F2B 10600678 IC50 = 89 nM T07806 CKH1P3 10601144 IC50 = 1200 nM T07806 CF74VT 10601619 Ki = 0.44 nM T07806 CC9B5J 10602052 IC50 = 66 nM T07806 C0LRY1 10612178 IC50 = 1348.96 nM T07806 CVYB63 10613373 Ki = 1 nM T07806 C1UVB3 10614906 IC50 = 310 nM T07806 CCVT79 10614907 IC50 = 145 nM T07806 CF5PK0 10617665 IC50 = 316.23 nM T07806 C8GFT6 10618751 Ki = 37 nM T07806 C06DSC 10620429 IC50 = 18 nM T07806 CWQ83M 10621020 IC50 = 209 nM T07806 CPF68U 10621021 IC50 = 11 nM T07806 CX09MP 10623434 IC50 = 540 nM T07806 CQO50M 10623614 IC50 = 25 nM T07806 C04NHF 10624003 IC50 = 2100 nM T07806 C8SN9G 10624768 Ki = 2.512 nM T07806 CN3H7E 10625408 IC50 = 140 nM T07806 CRB8C0 10635169 Ki = 425 nM T07806 C1MYD5 10640199 Ki = 21 nM T07806 C2FH3S 10643939 Ki = 13.6 nM T07806 C7R0EY 10643940 IC50 = 204.17 nM T07806 CLIA32 10644749 IC50 = 48 nM T07806 CQ98VE 10644750 IC50 = 18 nM T07806 CTM21V 10645471 IC50 = 170 nM T07806 C85DEQ 10645715 IC50 = 200 nM T07806 CDJ83U 10646873 IC50 = 58 nM T07806 CY7CU2 10646958 IC50 = 110 nM T07806 CPW89L 10646959 IC50 = 400 nM T07806 C0K2XA 10647181 IC50 = 25 nM T07806 C6PBY1 10647387 Ki = 0.32 nM T07806 CYDV92 10649124 Ki = 0.43 nM T07806 C6X0RT 10654938 Ki = 316 nM T07806 C4NW8J 10655811 Ki = 1995 nM T07806 C8W4FR 10663236 Ki = 53 nM T07806 CEVO29 10664203 Ki = 2 nM T07806 CA3E2W 10664878 IC50 = 1122.02 nM T07806 C5W6PY 10665156 Ki = 1.1 nM T07806 CNH98X 10665840 IC50 = 3801.89 nM T07806 CZ01DX 10667886 IC50 = 13 nM T07806 CTO51R 10670211 IC50 = 85 nM T07806 CB6YO4 10670534 IC50 = 5.3 nM T07806 C6XT1C 10670879 IC50 = 87 nM T07806 CR37GO 10671315 EC50 = 10000 nM T07806 CVA06U 10671996 IC50 = 260 nM T07806 C0U6ZS 10672840 Ki = 0.43 nM T07806 C4BS9A 10673329 Ki = 0.5012 nM T07806 C9U4LX 10679184 Ki > 10000 nM T07806 C8F1SI 10689227 IC50 = 325 nM T07806 C5FQ9T 10691904 Ki = 88 nM T07806 C9OHV5 10691928 IC50 = 260 nM T07806 COV35P 10693140 IC50 = 41 nM T07806 C2AI0W 10693206 IC50 = 33 nM T07806 CA3XK7 10693207 IC50 = 76 nM T07806 C4RN7E 10694177 IC50 = 1300 nM T07806 CSY6R8 10694810 IC50 = 5800 nM T07806 CSJ83Y 10694895 IC50 = 7200 nM T07806 CEIQ24 10695596 IC50 = 1600 nM T07806 CYI47N 10696275 IC50 = 170 nM T07806 CM31PB 10696930 EC50 = 0.09 nM T07806 COYX78 10709057 IC50 = 831.76 nM T07806 CE7DB9 10710400 Ki = 22 nM T07806 C97LJV 10714071 IC50 = 1202.26 nM T07806 CHW9D0 10716915 IC50 = 20 nM T07806 C3Y9FE 10717709 IC50 = 140 nM T07806 C4N7MI 10718668 IC50 = 165 nM T07806 CG6A0Q 10718714 IC50 = 140 nM T07806 C15RUN 10719202 IC50 = 102 nM T07806 CYHQ97 10719203 IC50 = 45 nM T07806 CL1UQ7 10719245 IC50 = 85 nM T07806 CM9H8J 10719448 IC50 = 60 nM T07806 C3F7XV 10719687 EC50 = 290 nM T07806 CX8U7Y 10719938 IC50 = 18 nM T07806 C2Y5UQ 10720175 IC50 = 9.3 nM T07806 CUS3R0 10720301 Ki = 0.11 nM T07806 C1FEW3 10733696 IC50 = 15 nM T07806 CAT6N3 10733823 IC50 = 7.4 nM T07806 CH1PV5 10739818 IC50 = 85 nM T07806 C3PBD8 10740531 IC50 = 125 nM T07806 C2IK5A 10741528 IC50 = 59 nM T07806 CIA9Z0 10741826 IC50 = 74 nM T07806 CX3FL8 10751317 Ki = 4.6 nM T07806 C61VBM 10757342 IC50 = 1513.56 nM T07806 CO0QF6 10759465 IC50 = 5100 nM T07806 CLBQ57 10764284 IC50 = 3900 nM T07806 CC49QS 10764869 IC50 = 130 nM T07806 CWYI16 10764998 IC50 = 35 nM T07806 CFXR10 10765655 IC50 = 28 nM T07806 C1I9OU 10766235 IC50 = 210 nM T07806 CNJ40K 10766277 IC50 = 140 nM T07806 CR2I0K 10766318 IC50 = 210 nM T07806 C2R0QI 10766319 IC50 = 150 nM T07806 CD7JC0 10766320 IC50 = 34 nM T07806 CJD70A 10766321 IC50 = 79 nM T07806 C8X2BM 10766570 EC50 = 1500 nM T07806 C48HGI 10767140 IC50 = 1000 nM T07806 CLDH19 10767244 IC50 = 8.9 nM T07806 CL5G7U 10768115 IC50 = 40 nM T07806 C54KOF 10768329 IC50 = 78 nM T07806 CP56UK 10774567 Ki = 5785 nM T07806 C5SP9E 10775772 Ki = 120 nM T07806 C9JW7S 10780344 IC50 = 93 nM T07806 CCB14F 10782381 IC50 = 6309.57 nM T07806 CZJO64 10782681 Ki = 40 nM T07806 CX70KH 10786335 Ki = 16.2 nM T07806 CB6Q0L 10786628 IC50 = 81 nM T07806 CP3V4H 10787240 IC50 = 2.7 nM T07806 CW5L3X 10787241 IC50 = 110 nM T07806 C7RC5Y 10788620 IC50 = 110 nM T07806 CK34DX 10788768 IC50 = 9.5 nM T07806 C78QWE 10789334 IC50 = 11 nM T07806 CC48LD 10789399 IC50 = 17 nM T07806 CSDI98 10789717 IC50 = 680 nM T07806 CKG19X 10790076 IC50 = 100 nM T07806 C8Y3TP 10791125 Ki = 1.4 nM T07806 CNUF06 10791244 EC50 = 0.19 nM T07806 C7GF8M 10791443 Ki = 2.512 nM T07806 CK9O3B 10802304 Ki = 1 nM T07806 C4UR8Q 10805740 IC50 = 275.42 nM T07806 CXY1Q0 10809674 Ki = 2.5 nM T07806 CU2QG3 10811007 IC50 = 47 nM T07806 CH94VG 10811801 IC50 = 93 nM T07806 CW1Y5T 10811964 IC50 = 89 nM T07806 CIL3O6 10812465 IC50 = 28 nM T07806 CZG3J2 10812592 IC50 = 49 nM T07806 CRN89V 10812693 IC50 = 3000 nM T07806 C8J2GW 10813272 IC50 = 230 nM T07806 CZT8S0 10813413 IC50 = 16 nM T07806 CA70HZ 10813769 IC50 = 150 nM T07806 C8NM9E 10814273 IC50 = 170 nM T07806 CW2LK3 10828231 Ki = 14 nM T07806 C7T1XC 10830159 Ki > 1000 nM T07806 C78FDC 10834908 IC50 = 575 nM T07806 CY15OU 10834909 IC50 = 22 nM T07806 C8MHZ9 10835110 Ki = 1584.89 nM T07806 CLE1W7 10835665 IC50 = 140 nM T07806 CMD47Q 10835928 IC50 = 24 nM T07806 CL2S9M 10836290 IC50 = 78 nM T07806 CF3W8J 10836301 IC50 = 59 nM T07806 C0MNA5 10836606 Ki = 0.5 nM T07806 C5L4HY 10836850 IC50 = 280 nM T07806 C30FNB 10836986 IC50 = 100 nM T07806 C2UJQ9 10837591 IC50 = 1300 nM T07806 CHCV53 10837853 EC50 = 5100 nM T07806 C83QOA 10837858 Ki = 0.2 nM T07806 CC8XL5 10838063 Ki = 0.38 nM T07806 C1ARP7 10838153 IC50 = 251 nM T07806 C1TI9X 10838622 IC50 = 350 nM T07806 C3IHO1 10838684 IC50 = 120 nM T07806 CCH9T7 10838923 Ki = 31.62 nM T07806 C1OL4F 10839082 IC50 = 66 nM T07806 C98RSP 10847427 Ki > 10000 nM T07806 C4V3RT 10848041 Ki = 1.6 nM T07806 C6D1CX 10852406 IC50 = 3890.45 nM T07806 CIG0Y6 10858566 Ki = 139 nM T07806 CPLT37 10870264 Ki = 210 nM T07806 C8HN1F 10872581 Ki = 270 nM T07806 C8OYI0 10891048 Ki = 2900 nM T07806 C84RHF 10896220 Ki = 11 nM T07806 C1RAP3 10904295 Ki = 80 nM T07806 C0Q7GV 10915350 Ki = 590 nM T07806 CL8AG5 10917920 Ki = 68 nM T07806 C2UZ8H 10917953 Ki = 220 nM T07806 CZN8J0 10925382 Ki = 1100 nM T07806 C5X1OQ 10926112 Ki = 1200 nM T07806 CWE3C9 10946905 Ki = 380 nM T07806 C7GHU5 10970604 Ki = 3.2 nM T07806 CN6BC3 10972931 Ki = 4.2 nM T07806 C5NRU3 10973768 Ki = 560 nM T07806 CJC9K4 11005810 IC50 = 3580 nM T07806 CJS79L 11011968 Ki = 1700 nM T07806 CN63RC 11016395 Ki = 5.9 nM T07806 CH9GU5 11016418 Ki = 480 nM T07806 CSU4T7 11024618 Ki = 6000 nM T07806 CX73TF 11035452 Ki = 150 nM T07806 C7BS5D 11038248 Ki = 20 nM T07806 C0ES3U 11038263 Ki = 20 nM T07806 C3G0FH 11046087 Ki = 1000 nM T07806 CG0J7X 11047115 Ki = 390 nM T07806 CC1YO2 11049209 Ki = 110 nM T07806 C5N9GT 11056946 Ki = 390 nM T07806 CFJG64 11059058 IC50 = 708 nM T07806 C0FT4D 11067619 Ki = 820 nM T07806 CUJ4W7 11071135 Ki = 100 nM T07806 CM2BD4 11092112 Ki = 360 nM T07806 CE42CZ 11092142 Ki = 6.5 nM T07806 C0G3WS 11098166 Ki = 14 nM T07806 CRU3M5 11110452 Ki = 1000 nM T07806 C4VRT9 11111280 Ki = 750 nM T07806 CTBF50 11120893 Ki = 930 nM T07806 C6G9KQ 11123573 Ki = 31 nM T07806 CPA0G8 11145333 Ki = 76 nM T07806 C6CL1Y 11178830 Ki = 398.11 nM T07806 C9N5QU 11200511 Ki = 15 nM T07806 CPX23W 11209208 IC50 > 10000 nM T07806 C6D1MZ 11223004 Ki = 88 nM T07806 C6MI9K 11235335 Ki = 316.23 nM T07806 C90WSG 11248705 Ki = 1584.89 nM T07806 CAPX71 11259254 Ki = 199.53 nM T07806 C8JW3Z 11260311 Ki > 1000 nM T07806 CO25MT 11270107 Ki = 79.43 nM T07806 C27GXZ 11277680 IC50 > 10000 nM T07806 C57GTA 11299968 IC50 > 10000 nM T07806 C9BLC7 11304596 Ki = 1.995 nM T07806 CJS9C0 11304851 IC50 > 3200 nM T07806 CI79LV 11307899 Ki = 3.162 nM T07806 CUXZ91 11311148 IC50 > 10000 nM T07806 C2GZD3 11311204 IC50 > 10000 nM T07806 CTN62X 11328382 Ki = 2.512 nM T07806 CBV52J 11384146 Ki = 4.3 nM T07806 CF4OX6 11397149 Ki = 3.162 nM T07806 CGV14H 11402988 Ki = 23 nM T07806 CCA2X4 11407766 Ki < 10000 nM T07806 CKL9J7 11419978 Ki = 3.162 nM T07806 CG4ST6 11464355 Ki = 398.11 nM T07806 CCGF98 11476072 Ki = 316.23 nM T07806 C38QFE 11530118 IC50 > 10000 nM T07806 CQ08DH 11539632 IC50 = 0.2 nM T07806 C9VC7O 11551780 IC50 > 10000 nM T07806 CNH1K4 11568826 Ki = 2.5 nM T07806 C6JC2T 11580039 IC50 > 10000 nM T07806 C6D1MA 11584660 Ki > 501.19 nM T07806 CKWA60 11591924 Ki = 3.162 nM T07806 CGX8F6 11596869 Ki > 3580000 nM T07806 CNEV03 11626724 IC50 = 83 nM T07806 CKO3M0 11647963 IC50 = 47 nM T07806 CX7FR8 11655728 Ki = 0.7943 nM T07806 C4L7TV 11662592 Ki = 9.7 nM T07806 C75URP 11668825 IC50 = 32 nM T07806 CHK5I2 11712756 Ki = 1.259 nM T07806 CX9VH0 11720815 Ki = 1 nM T07806 C74LAD 11723305 Ki = 82 nM T07806 CZE25U 11725335 Ki = 373 nM T07806 CSL02Y 11726413 Ki = 279 nM T07806 C3T9XB 11727140 Ki = 640 nM T07806 CL97KG 11728004 Ki = 32 nM T07806 CD49YX 11740144 Ki = 14 nM T07806 CPZ5N7 11740280 Ki = 40 nM T07806 C6B4YJ 11743042 Ki = 224 nM T07806 CPG15O 11743399 IC50 > 1000 nM T07806 CYV02C 11747350 Ki = 910 nM T07806 CG2WS6 11759467 Ki = 330 nM T07806 CK1C4D 11774585 Ki = 251.19 nM T07806 CJ3G6W 11777940 Ki = 312 nM T07806 CB3NF0 11778645 Ki = 219 nM T07806 CYZP79 11794624 Ki = 125.89 nM T07806 C7EWM8 11794750 IC50 = 12 nM T07806 CCR26G 11795333 IC50 = 23 nM T07806 C4U5IW 11795525 IC50 = 78 nM T07806 CV5UF3 11795644 IC50 = 41 nM T07806 CC69IB 11796081 IC50 = 260 nM T07806 C6TM2A 11796257 Ki = 6.31 nM T07806 CDJ7T1 11796806 IC50 = 140 nM T07806 C7R9MY 11796807 IC50 = 305 nM T07806 C0DTJ5 11796808 IC50 = 575 nM T07806 CAMY96 11797158 Ki = 0.16 nM T07806 CIK15Y 11797562 IC50 = 160 nM T07806 C3U7IY 11797644 IC50 = 50 nM T07806 CN2BP0 11797998 Ki = 0.1 nM T07806 CY75KM 11797999 Ki = 1.7 nM T07806 CQ35ZC 11798094 IC50 = 2.4 nM T07806 CFMK96 11798502 IC50 = 282 nM T07806 C9AT7N 11798621 IC50 = 85 nM T07806 CS19AU 11800592 Ki = 0.27 nM T07806 CUI5G6 11809037 Ki = 25 nM T07806 CF9T0I 11810310 Ki = 1600 nM T07806 C2R3GJ 11812916 Ki = 45 nM T07806 CL1J7U 11822996 Ki = 610 nM T07806 CVW4B5 11824522 Ki = 310 nM T07806 CJ49VT 11826976 Ki = 14 nM T07806 CE1QZ8 11827039 Ki = 2.8 nM T07806 CXLW54 11948707 Ki = 228 nM T07806 C8JQL7 11957735 IC50 > 10000 nM T07806 CR7TS2 12361789 Ki > 1000 nM T07806 C2QAC7 12406830 Ki = 1430 nM T07806 CVSW49 12987128 Ki > 10000 nM T07806 CC0ZK7 13096730 Ki = 349 nM T07806 CI5N4L 13520547 Ki = 470 nM T07806 C5J7WY 14519851 Ki = 100 nM T07806 CM1N9P 14519863 Ki = 2675 nM T07806 CWK85F 14519865 Ki = 750 nM T07806 C87QBZ 14547414 Ki = 228 nM T07806 CJG80D 14547415 Ki = 1690 nM T07806 CQ7I1H 14566707 Ki = 290 nM T07806 CTSI74 14639163 Ki = 1630 nM T07806 CYW76P 14742527 Ki > 1000 nM T07806 C4R5JF 15516681 IC50 = 27 nM T07806 C62NLP 15516682 IC50 = 19 nM T07806 CX0P5R 15516683 IC50 = 61 nM T07806 C1SR0O 16071847 Ki > 5000 nM T07806 CZ1WJ4 16117151 Ki = 1659 nM T07806 CM32ZX 16117153 Ki > 5000 nM T07806 CXTB90 16117279 Ki = 2726 nM T07806 C1F2LS 16118795 Ki > 5000 nM T07806 C69VDS 16118923 Ki > 5000 nM T07806 CZ2IS9 16660294 Ki > 10000 nM T07806 C4YMP1 16725956 Ki > 1000 nM T07806 C0T9ZY 17947861 Ki = 5.012 nM T07806 CHXQ26 18366015 IC50 = 562.34 nM T07806 CUJ1C8 18691541 IC50 = 18.2 nM T07806 CI1DQ5 18691565 IC50 = 97.72 nM T07806 CP07ZI 18691566 IC50 = 32.36 nM T07806 CE5GD1 18975338 IC50 = 360 nM T07806 CP8S5X 18975369 IC50 = 19 nM T07806 CYJ48A 19066163 Ki = 1.3 nM T07806 C0BE1M 19066188 Ki = 18 nM T07806 CV5FR6 19066200 Ki = 8.4 nM T07806 C4RU6O 19066201 Ki = 2 nM T07806 CN96TB 19066203 Ki = 1.8 nM T07806 C60SWJ 19066205 Ki = 8 nM T07806 C5MS9T 19066235 Ki = 40 nM T07806 CQ3JL0 19956256 IC50 = 2691.53 nM T07806 C7T8JC 19958494 Ki > 10000 nM T07806 C6LI5E 19958507 Ki > 10000 nM T07806 CT1C6U 20255884 Ki = 10240 nM T07806 C3T5HF 21509921 Ki = 1348.96 nM T07806 CT7XG9 21830793 Ki = 643 nM T07806 CYH4J9 22002244 Ki = 70.3 nM T07806 CBN84K 22065997 Ki > 10000 nM T07806 CWXC93 22067856 Ki = 3450 nM T07806 CE65DB 22115679 Ki < 1 nM T07806 CL20SZ 22184640 Ki = 170 nM T07806 CY7TL3 22184642 Ki > 1000 nM T07806 CWY17R 22184652 Ki = 0.9 nM T07806 C2Z0BJ 22326660 Ki = 1000 nM T07806 CD80PB 22326688 Ki = 3.981 nM T07806 CJ3P6O 22326704 Ki = 31.62 nM T07806 C5SI3U 22464564 Ki = 319.6 nM T07806 CJ6WF3 22464606 Ki = 3.8 nM T07806 CA5BY9 22464614 Ki = 50.2 nM T07806 CQB94R 22464634 Ki = 36.6 nM T07806 CAZ23L 22464649 Ki = 0.5 nM T07806 CJCY98 22464720 Ki = 1.7 nM T07806 CB97XC 22464804 Ki = 5.4 nM T07806 C9MB7K 22464806 Ki = 116.4 nM T07806 C7DXE6 22464831 Ki = 3.5 nM T07806 C76FEA 22464842 Ki = 1.4 nM T07806 CRU1N2 22611622 Ki = 390 nM T07806 CD4JS0 23274477 Ki = 255 nM T07806 CR1F5X 23374587 IC50 = 4.4 nM T07806 C93XHZ 23533306 Ki = 9.3 nM T07806 CCKZ73 23533322 Ki = 3.5 nM T07806 C6EK2V 23533328 Ki = 392 nM T07806 C6WNZ9 23533329 Ki = 292 nM T07806 C60NCW 24755624 Ki < 3162.28 nM T07806 C6GBU8 24762221 EC50 = 199.53 nM T07806 CD7CV6 24771120 Ki > 2000 nM T07806 CJ4RO1 24804774 EC50 = 398.11 nM T07806 CK84BF 24804775 Ki = 0.7943 nM T07806 C1Z3OQ 24804941 Ki > 1000 nM T07806 C6AE2U 24804942 Ki > 1000 nM T07806 C1ZYM4 24804943 Ki > 1000 nM T07806 CDC91N 24839550 Ki < 10000 nM T07806 CY21RE 24841480 Ki = 2200 nM T07806 CF8I9P 24845776 Ki < 6309.57 nM T07806 C93JWY 24865538 Ki = 251.19 nM T07806 C5F2VL 24865539 Ki = 501.19 nM T07806 CW9N1Z 24865540 Ki = 1258.93 nM T07806 C8PXH7 24865541 Ki = 1584.89 nM T07806 CN5VB4 24865542 Ki = 50.12 nM T07806 CPF5E2 24865543 Ki = 39.81 nM T07806 CGDV58 24865724 Ki = 100 nM T07806 C3HK0J 24865725 Ki = 1.995 nM T07806 C5TX3M 24865726 Ki = 12.59 nM T07806 C0O6FX 24865727 Ki = 12.59 nM T07806 CER0O4 24881201 Ki = 16 nM T07806 C5ZK1C 24881202 Ki = 1.3 nM T07806 C1OF5Z 24881203 Ki = 0.79 nM T07806 C02XDI 24881204 Ki = 0.5 nM T07806 C82DUO 24881264 Ki = 0.81 nM T07806 CIA98Y 24881550 Ki = 103 nM T07806 CMS4W9 24881551 Ki > 1000 nM T07806 CDW36L 24881552 Ki > 10000 nM T07806 C8OGB4 24881617 Ki = 100 nM T07806 CFMS90 24881618 Ki = 126 nM T07806 CUF79T 24881619 Ki = 126 nM T07806 C18SOA 24881686 Ki = 32 nM T07806 CCQY75 24881687 Ki = 453 nM T07806 C49DNT 24881688 Ki > 1000 nM T07806 CJSL82 24881689 Ki = 0.76 nM T07806 CXA24K 24881752 Ki = 1.3 nM T07806 CZ5Q6P 24881753 Ki = 0.1 nM T07806 C4FWN1 24881754 Ki = 0.58 nM T07806 COU24N 24882192 Ki > 10000 nM T07806 C43RTZ 24882193 Ki = 79 nM T07806 C8B4YF 24882266 Ki = 38 nM T07806 CNO84Q 24882267 Ki > 10000 nM T07806 CK6R9A 24882268 Ki = 18 nM T07806 C6L7KS 24887518 Ki < 3162.28 nM T07806 C1VRJ3 25014630 IC50 = 2200 nM T07806 CCTG60 25022506 Ki < 3162.28 nM T07806 CYJ5G1 25067564 Ki = 6040 nM T07806 C4B0FU 25070577 IC50 = 610 nM T07806 CM2T9Y 25263297 Ki > 2000 nM T07806 CFJM71 25263302 Ki = 1800 nM T07806 CA58DL 41305446 Ki = 8594 nM T07806 CXZH39 44138098 Ki = 1 nM T07806 CUOD42 44138104 Ki = 1.585 nM T07806 C92CVD 44214329 Ki = 17 nM T07806 CYN83E 44214559 IC50 = 13 nM T07806 CCP37Q 44267158 IC50 < 100000 nM T07806 CFEI56 44267161 IC50 = 7413.1 nM T07806 CHU4L9 44267168 IC50 = 1584.89 nM T07806 CIZ5W7 44267181 IC50 = 22908.68 nM T07806 CFE12G 44267205 IC50 = 35481.34 nM T07806 C5CPZ7 44267215 IC50 = 138038.43 nM T07806 CC2OD4 44278111 Ki > 10000 nM T07806 CRMA84 44278114 Ki > 10000 nM T07806 CF0Y4M 44278115 Ki > 10000 nM T07806 C08LZS 44279525 Ki = 0.76 nM T07806 C1OI7G 44279549 Ki = 0.7 nM T07806 CFWE96 44279550 Ki = 2.56 nM T07806 C7DR8P 44279889 Ki = 2.1 nM T07806 CS3HX6 44292365 Ki = 15.5 nM T07806 C32ARH 44292367 Ki = 118 nM T07806 C1Y0JR 44292375 Ki = 10.4 nM T07806 CZL18K 44310169 Ki = 2024 nM T07806 C5Q1VH 44311908 Ki = 3735 nM T07806 CYI2D8 44311953 Ki > 10000 nM T07806 CS9Z7Q 44323506 IC50 = 220 nM T07806 CS7NA2 44337678 Ki = 0.8 nM T07806 CU4F3W 44337731 Ki = 11 nM T07806 CUT24A 44338900 Ki = 59 nM T07806 CL2KT5 44339071 Ki = 63 nM T07806 CT8FG6 44339072 Ki = 52 nM T07806 C9AP7L 44341609 IC50 = 89 nM T07806 CW2MP5 44341625 IC50 = 30 nM T07806 C5S2NC 44341637 IC50 = 55 nM T07806 C0WZJ1 44341657 IC50 = 57 nM T07806 CIC09X 44341707 IC50 = 27 nM T07806 C8B4XQ 44341783 IC50 = 340 nM T07806 CLD14T 44341798 IC50 = 85 nM T07806 CME4B2 44342506 Ki = 1.5 nM T07806 CVI4J5 44342507 Ki = 39 nM T07806 CX8LV0 44342508 Ki = 3.8 nM T07806 C3I7YQ 44342518 Ki = 3.8 nM T07806 CAUL48 44342705 Ki = 14 nM T07806 CNSF41 44342722 Ki = 4.8 nM T07806 CIA3M0 44342727 Ki = 14 nM T07806 C7OQD9 44342767 Ki = 5.8 nM T07806 CQV5X1 44342783 Ki = 13 nM T07806 CC08TZ 44342784 Ki = 1.5 nM T07806 C9KGS3 44342785 Ki = 2.4 nM T07806 CBGP96 44342823 Ki = 11 nM T07806 C1URA6 44342830 Ki = 4.2 nM T07806 C9K5VL 44342969 Ki = 17 nM T07806 C7YS8F 44342993 Ki = 3.2 nM T07806 CPWJ26 44343212 Ki < 10000 nM T07806 C9Y8WE 44344504 IC50 = 568 nM T07806 CX3ZL5 44351656 Ki = 0.14 nM T07806 CUXH48 44352308 Ki = 1060 nM T07806 CS3J6N 44363580 Ki > 100 nM T07806 C3LKN1 44364048 Ki = 316.23 nM T07806 CVS5L1 44364110 IC50 = 300 nM T07806 C0AJ1Z 44376262 Ki = 44 nM T07806 C6FLR4 44376263 Ki = 82 nM T07806 CS32NH 44376272 Ki = 68 nM T07806 C9S8OK 44376278 Ki = 64 nM T07806 COT84H 44376280 Ki = 140 nM T07806 C89EPR 44376282 Ki = 36 nM T07806 CHFE56 44376283 Ki = 170 nM T07806 C94ACX 44376362 Ki = 760 nM T07806 C3JEU0 44376363 Ki = 95 nM T07806 C0W7LR 44376383 Ki = 32 nM T07806 C86TNU 44376395 Ki = 58 nM T07806 CTF4O0 44376491 Ki = 410 nM T07806 CRE24Q 44376492 Ki = 110 nM T07806 CKDU28 44376494 Ki = 130 nM T07806 C8C2KA 44376516 Ki = 40 nM T07806 CQVX74 44376541 Ki = 65 nM T07806 CJ90UO 44376588 Ki = 140 nM T07806 CL7O3J 44376722 Ki = 63 nM T07806 C2MAB6 44376723 Ki = 38 nM T07806 C0U9RL 44383728 Ki = 476 nM T07806 C5RYQ7 44383729 Ki = 107 nM T07806 CM0T9D 44383737 Ki = 9.9 nM T07806 CV4C3R 44383738 Ki = 113 nM T07806 CIS4L0 44394222 Ki = 12 nM T07806 C9K4SC 44395787 Ki = 2400 nM T07806 C93XHA 44395809 Ki = 440 nM T07806 C9A4NM 44395832 Ki = 260 nM T07806 C4B0OI 44397588 Ki = 630.96 nM T07806 C5FP0R 44397589 Ki = 630.96 nM T07806 CE3G8U 44397670 Ki = 316.23 nM T07806 C1KA3F 44400359 Ki = 100 nM T07806 C9THQ3 44402868 Ki = 3.981 nM T07806 C1EI5Q 44402869 Ki = 31.62 nM T07806 CV0PC9 44402870 Ki = 3.981 nM T07806 CV15IH 44402871 Ki = 7.943 nM T07806 CD20SO 44402874 Ki = 12.59 nM T07806 CM45GD 44402875 Ki = 19.95 nM T07806 CG1WU9 44402876 Ki = 1.995 nM T07806 C6WNI4 44402877 Ki = 3.162 nM T07806 CDL1F6 44402878 Ki = 50.12 nM T07806 CLR72M 44402879 Ki = 1.995 nM T07806 CZL9Y8 44402880 Ki = 3.162 nM T07806 CHU6W5 44402881 Ki = 3.981 nM T07806 C8ZJ7W 44402882 Ki = 2.512 nM T07806 C6M8WP 44402883 Ki = 2.512 nM T07806 CKX16M 44402884 Ki = 2.512 nM T07806 CHG01P 44402885 Ki = 0.631 nM T07806 CD37FS 44402886 Ki = 3.162 nM T07806 CI4MO9 44402887 Ki = 1.585 nM T07806 CX89BK 44402888 Ki = 7.943 nM T07806 CSDV68 44402893 Ki = 7.943 nM T07806 CY4FD0 44402894 Ki = 5.012 nM T07806 CRWN42 44402895 Ki = 5.012 nM T07806 C1B4QL 44403095 Ki = 1.82 nM T07806 C1YL7Z 44403098 Ki = 38.3 nM T07806 CFV98A 44403101 Ki = 13.7 nM T07806 C6OY9S 44403102 Ki = 28.4 nM T07806 CH4SX6 44403105 Ki = 16.7 nM T07806 C12FIH 44403106 Ki = 9.68 nM T07806 CI0WG5 44404225 Ki = 0.3162 nM T07806 C7FAW3 44404229 Ki = 0.5012 nM T07806 C0MXR4 44404230 Ki = 15.85 nM T07806 C7OD6Q 44404236 Ki = 1.259 nM T07806 C5W2KR 44404240 Ki = 0.2512 nM T07806 CI50CY 44404241 Ki = 0.7943 nM T07806 CF69DU 44404244 Ki = 1.995 nM T07806 CE0NI6 44404245 Ki = 15.85 nM T07806 CLW3P7 44404249 Ki = 1 nM T07806 CF8LN5 44404253 Ki = 2.512 nM T07806 C3LI6E 44404258 Ki = 1.585 nM T07806 C2NH8G 44404260 Ki = 3.981 nM T07806 C7R5HU 44404264 Ki = 7.943 nM T07806 CVTZ13 44404268 Ki = 1 nM T07806 C18ISW 44404272 Ki = 1.995 nM T07806 C4LKC1 44404394 Ki = 11.3 nM T07806 C3EJ4G 44404396 Ki = 18.1 nM T07806 C7W3BP 44405573 Ki = 1.1 nM T07806 CV9IR7 44405574 Ki = 1.1 nM T07806 CFG72V 44405575 Ki = 1.2 nM T07806 C8WSZ2 44405586 Ki = 2.5 nM T07806 CEJ0C3 44405587 Ki = 5.4 nM T07806 C4DK0U 44405655 Ki = 11.9 nM T07806 C28WCH 44405665 Ki = 42.3 nM T07806 CS7ZD5 44405666 Ki = 0.5 nM T07806 CIH9J0 44405669 Ki = 0.4 nM T07806 CVZO38 44405677 Ki = 3.3 nM T07806 CMK32Z 44405701 Ki = 1.7 nM T07806 CZK5L6 44405702 Ki = 0.9 nM T07806 CO7G3W 44405725 Ki = 0.5 nM T07806 CU1VL9 44405726 Ki = 4.9 nM T07806 CO1P3W 44405730 Ki = 0.1 nM T07806 CG87PW 44409290 Ki > 720 nM T07806 CV5MY8 44422352 Ki = 35 nM T07806 C6AV7K 44422357 Ki > 1000 nM T07806 CL59HA 44431531 Ki = 281 nM T07806 C6JK5A 44431532 Ki = 103 nM T07806 C5LNH6 44431533 Ki = 91 nM T07806 CLX73C 44431534 Ki > 1000 nM T07806 CCV62B 44431535 Ki > 1000 nM T07806 C4P5XG 44431536 Ki = 21 nM T07806 CYPR70 44431537 Ki = 15 nM T07806 CY9IK3 44438461 Ki = 31 nM T07806 C6W2EZ 44438462 Ki = 414 nM T07806 C9IFR5 44438464 Ki = 1490 nM T07806 CLWE65 44438469 Ki > 300 nM T07806 CKZF16 44439165 Ki = 1995.26 nM T07806 CA4HZ3 44439167 Ki = 630.96 nM T07806 CT0C4I 44443093 Ki = 7.943 nM T07806 C8E1AC 44443094 Ki = 25.12 nM T07806 CZ6BK9 44443095 Ki = 31.62 nM T07806 CV5T2C 44443096 Ki = 31.62 nM T07806 CT1S6L 44443097 Ki = 31.62 nM T07806 CF1V8O 44443098 Ki = 63.1 nM T07806 CHZ48Q 44443101 Ki = 25.12 nM T07806 CQ53TV 44443130 Ki = 0.1995 nM T07806 CEZ6U8 44443131 Ki = 1.585 nM T07806 CN4XZ6 44443132 Ki = 1.585 nM T07806 CM8AY5 44444556 Ki = 12.59 nM T07806 CW9LC3 44444557 Ki = 1995.26 nM T07806 CZL97F 44455426 Ki = 1846 nM T07806 C12XGE 44456400 Ki > 10000 nM T07806 CP2F5J 44460810 Ki = 186 nM T07806 C6GHE9 44460826 Ki = 200 nM T07806 CXB7G1 44461149 Ki = 155 nM T07806 CZ5E2H 44461168 Ki > 1000 nM T07806 C8YD0T 44461234 Ki > 1000 nM T07806 CJAI80 44461247 Ki = 310 nM T07806 C3R5WE 44461248 Ki = 96 nM T07806 C9TXL1 44461249 Ki = 131 nM T07806 CI0RQ9 44461251 Ki > 1000 nM T07806 CQ4S9I 44461266 Ki > 1000 nM T07806 CO0ZT7 44461293 Ki > 1000 nM T07806 C6UTB1 44461297 Ki = 210 nM T07806 C9GJ3W 44461298 Ki = 155 nM T07806 C2ZH0I 44461300 Ki > 1000 nM T07806 CCT61W 44461306 Ki = 316 nM T07806 C09MBT 44461308 Ki > 1000 nM T07806 CJHL27 44461335 Ki > 1000 nM T07806 CT06WG 44461336 Ki > 1000 nM T07806 CB8C2D 44461416 Ki > 1000 nM T07806 CIN15X 44461425 Ki = 210 nM T07806 CHL8S2 44461443 Ki = 73 nM T07806 C2IDH4 44461586 Ki > 1000 nM T07806 C3D4HR 44537940 Ki > 5000 nM T07806 CJ7U3K 44554227 Ki > 5000 nM T07806 CM0I1P 44554393 Ki > 5000 nM T07806 CNHA47 44554395 Ki = 3624 nM T07806 CB23PH 44560995 Ki = 60 nM T07806 CZO5Y8 44580740 Ki = 1.259 nM T07806 C4N6PM 44580741 Ki = 7.943 nM T07806 C0XVL5 44580783 Ki = 0.7943 nM T07806 C4SD7P 44580784 Ki = 125.89 nM T07806 CNOU35 44581235 Ki = 79.43 nM T07806 CO6E5K 44581260 Ki = 31.62 nM T07806 CS6HG9 44581603 Ki = 6.31 nM T07806 C1HAQ2 44581604 Ki = 158.49 nM T07806 C5NS6H 44581972 Ki = 524.81 nM T07806 CK8Z1P 44581973 Ki = 776.25 nM T07806 C3UQ9Z 44581974 Ki = 588.84 nM T07806 CRCH48 44582675 Ki = 884 nM T07806 CEJ4R8 44582676 Ki = 2174 nM T07806 CZGP86 44582677 Ki > 10000 nM T07806 C5QB4K 44582678 Ki = 4886 nM T07806 C01RCI 44582705 Ki = 3359 nM T07806 CXL25V 44582706 Ki > 10000 nM T07806 C8MR1X 44582707 Ki > 10000 nM T07806 C4IT1N 44582708 Ki > 10000 nM T07806 C17LZR 44585926 Ki > 1000 nM T07806 CCU63Y 44585927 Ki > 1000 nM T07806 C5PG1H 44585928 Ki > 1000 nM T07806 CY1LE7 44585929 Ki > 1000 nM T07806 CMY8N9 44585945 Ki > 1000 nM T07806 C0S5ER 44585946 Ki > 1000 nM T07806 CSF39B 44588698 Ki > 10000 nM T07806 C7SKM1 44588720 Ki = 199.53 nM T07806 CI6SO1 44588721 Ki = 50.12 nM T07806 CB14UQ 44588722 Ki = 316.23 nM T07806 CNK64D 44588742 Ki = 398.11 nM T07806 CAT73D 44588743 Ki > 2511.89 nM T07806 C6DK3E 44588744 Ki > 10000 nM T07806 C9BO7K 44588745 Ki = 25.12 nM T07806 CD2CU8 44588771 Ki > 5011.87 nM T07806 CDIQ25 44588772 Ki = 630.96 nM T07806 C4EH6O 44592207 Ki = 31.62 nM T07806 CZ5I1N 44592208 EC50 = 6.31 nM T07806 CKM8T7 44592209 Ki = 3.981 nM T07806 CDJ32U 44592249 Ki = 5.012 nM T07806 CS2FL4 44592250 Ki = 5.012 nM T07806 CL17WU 44592251 Ki = 6.31 nM T07806 CJCL64 44592252 Ki = 15.85 nM T07806 CM0I3E 44592294 Ki = 2.512 nM T07806 CQ04EG 44592295 Ki = 15.85 nM T07806 C65XQL 44592296 Ki = 2.512 nM T07806 CEB2S1 44592297 Ki = 1.995 nM T07806 CP51QS 44592332 EC50 = 63.1 nM T07806 CD2Z4J 44592333 EC50 = 25.12 nM T07806 C7NCT2 44592334 Ki = 794.33 nM T07806 CHY20X 44592335 Ki = 158.49 nM T07806 C5H7XK 44592371 EC50 = 15.85 nM T07806 CZ0W1I 44593711 Ki = 39.81 nM T07806 CVCQ85 45104767 Ki = 0.4266 nM T07806 C4BP9Z 45104862 Ki = 0.955 nM T07806 C98UOH 45260312 Ki < 10000 nM T07806 C6Y0LZ 45260341 Ki < 10000 nM T07806 CHLR80 45260355 Ki = 158.49 nM T07806 C31CPA 45260363 Ki = 1000 nM T07806 CNQ7G1 45260372 Ki = 158.49 nM T07806 C2YL4K 45260377 Ki = 100 nM T07806 C7LRZ1 45260417 Ki = 6309.57 nM T07806 CRV8Z4 46232642 Ki = 9.3 nM T07806 C1JSH9 46899637 Ki = 1.585 nM T07806 C3MSL0 46899638 Ki = 1.585 nM T07806 CV3LP2 46899639 Ki = 1 nM T07806 CGHZ15 46899640 Ki = 1.585 nM T07806 CN9FC3 46900150 Ki = 1.585 nM T07806 C40ZJO 46900451 Ki = 1.585 nM T07806 CNC02A 46900453 Ki = 1.995 nM T07806 CTCH14 46900455 Ki = 1 nM T07806 CP41AQ 46900457 Ki = 1 nM T07806 CR3L4I 46900459 Ki = 0.7943 nM T07806 CK17PA 46900606 Ki = 2.512 nM T07806 CQ2K1C 46900608 Ki = 7.943 nM T07806 C5ZT1B 46900610 Ki = 1.259 nM T07806 C1NAX4 46900612 Ki = 1 nM T07806 CT0SQ2 46900614 Ki = 2.512 nM T07806 CXD9S3 46900776 Ki = 0.631 nM T07806 C8I7SJ 46900778 Ki = 1.585 nM T07806 C7QDM9 46900782 Ki = 2.512 nM T07806 C15FMY 46900954 Ki = 0.5012 nM T07806 C8W1FU 46900956 Ki = 0.631 nM T07806 CH35BV 46900958 Ki = 1.995 nM T07806 CO69SV 46905266 Ki = 199 nM T07806 C1QV6Y 46945444 Ki > 10000 nM T07806 CV93BN 46945445 Ki > 10000 nM T07806 C0H1AC 46945446 Ki = 1571 nM T07806 CLP8O6 46945447 Ki > 10000 nM T07806 C2LZJ0 49783209 Ki = 820 nM T07806 C57SMG 49783415 Ki > 10000 nM T07806 C0TG6I 49783419 Ki > 10000 nM T07806 C4HIZ8 49799868 Ki = 387 nM T07806 CR40BA 49836386 IC50 = 340 nM T07806 C0M5XC 49836496 IC50 = 500 nM T07806 C3OHN0 49850566 Ki = 3.981 nM T07806 C4R2YS 49850567 Ki = 1.259 nM T07806 CSGQ38 49850568 Ki = 3.162 nM T07806 C8P5KH 49850569 Ki = 1.995 nM T07806 C07JTU 49850570 Ki = 1.259 nM T07806 C6FP9W 49850571 Ki = 1.995 nM T07806 C3BVK5 49850668 Ki = 3.981 nM T07806 C6P3RH 49850669 Ki = 1 nM T07806 CGYT84 49850670 Ki = 3.981 nM T07806 C6Y3DW 49850671 Ki = 3.162 nM T07806 CK68QR 49850672 Ki = 0.5012 nM T07806 CI6O9A 49850673 Ki = 1.259 nM T07806 COFA76 49850768 Ki = 12.59 nM T07806 C4IX5R 49850769 Ki = 39.81 nM T07806 CXLT59 49850770 Ki = 31.62 nM T07806 C48DOX 49850771 Ki = 39.81 nM T07806 CN5XR1 49850772 Ki = 1.585 nM T07806 CR4EZ0 49850870 Ki = 0.7943 nM T07806 C5K4EC 49850872 Ki = 0.5012 nM T07806 C8AW0R 49850874 Ki = 2.512 nM T07806 CB2K6D 49850877 Ki = 3.162 nM T07806 C85KPE 49850980 Ki = 5.012 nM T07806 C5U3YD 49850982 Ki = 3.981 nM T07806 CV62IZ 49850984 Ki = 1.585 nM T07806 CED9V6 49852000 Ki = 1.995 nM T07806 CA0PW5 49852001 Ki = 1.259 nM T07806 C5S6BY 49852002 Ki = 1.585 nM T07806 C13ZTD 49852003 Ki = 1.995 nM T07806 CK17IE 49852105 Ki = 7.943 nM T07806 C2RY0J 50878551 Ki = 128.82 nM T07806 C1W6TV 50898777 Ki > 10000 nM T07806 CXMZ73 50898778 Ki > 10000 nM T07806 C67IRJ 50908804 Ki > 1000 nM T07806 CLOB24 50908805 Ki > 1000 nM T07806 CE4KP1 51050257 Ki > 10000 nM T07806 CRI12K 52942395 Ki = 13 nM T07806 CX9AF4 52942551 Ki = 0.631 nM T07806 CR0G5U 52942644 Ki = 1.995 nM T07806 CCF97B 52943811 EC50 = 501.19 nM T07806 C2FG9O 52943861 Ki = 31.62 nM T07806 C9G4CI 52943891 Ki > 1000 nM T07806 CCVP06 52944840 Ki = 398.11 nM T07806 CJ49MX 52946290 EC50 = 316.23 nM T07806 CK5ER0 52947414 Ki = 0.7943 nM T07806 CAVB03 52947615 Ki = 0.7943 nM T07806 C1HRK4 52947622 Ki = 316.23 nM T07806 C4ZC1K 52948697 EC50 = 63.1 nM T07806 CGY45S 53248361 Ki = 121 nM T07806 CE9L8G 53248365 Ki = 272 nM T07806 CCY98O 56935645 Ki = 120 nM T07806 C1TC7Q 56963799 Ki > 10000 nM T07806 CU4FW8 57397383 IC50 = 10000 nM T07806 C1LEH8 67268994 Ki > 10000 nM T07806 CLS9Y8 67650695 IC50 = 170 nM T07806 C63DCO 67650716 IC50 = 220 nM T07806 CP9V6A 69836292 Ki = 15.85 nM T07806 C3XNC2 71450247 Ki > 10000 nM T07806 C8P9EA 71450983 IC50 = 220 nM T07806 C4NDR3 71452382 Ki > 10000 nM T07806 C6ZWV2 71452383 Ki > 10000 nM T07806 CYK20Z 71452384 Ki = 956 nM T07806 C2ZGV6 71452688 Ki = 1617 nM T07806 CAQF34 71455625 Ki > 10000 nM T07806 CMJ1O9 71457409 Ki > 10000 nM T07806 CVI7S2 71457690 Ki = 7137 nM T07806 CPO82B 71458050 Ki = 7.943 nM T07806 CS83IF 71459269 Ki > 10000 nM T07806 CK5T4P 71459604 Ki = 6306 nM T07806 CG0WO9 71459954 Ki = 9.3 nM T07806 CJT49M 71459969 IC50 = 13 nM T07806 C63YLA 71461049 Ki > 10000 nM T07806 CJD96I 71461050 Ki > 10000 nM T07806 C6VL5X 71461632 Ki = 0.2 nM T07806 C85EAM 71461714 IC50 = 300 nM T07806 C4P3JU 71462776 Ki > 10000 nM T07806 C3GUQ2 71462777 Ki > 10000 nM T07806 C1Y9IC 71463063 Ki > 10000 nM T07806 C8Z0NM 72550642 Ki = 131 nM T07806 CL6W2Q 72550645 Ki = 7 nM T07806 C78LYM 72698087 Ki > 10000 nM T07806 C63HPK 72698088 Ki > 10000 nM T07806 CC6Q5R 72771081 Ki < 100 nM T07806 CC65OA 73213195 Ki = 707.95 nM T07806 CW83DK 73213196 Ki = 1218 nM T07806 CCV91B 73346042 Ki = 411 nM T07806 CK0HR9 73346334 Ki > 10000 nM T07806 C8GQK9 73350823 Ki = 700 nM T07806 C2E7QW 75201901 Ki = 9300 nM T07806 C8IDL3 75306277 Ki = 316.23 nM T07806 C4P8QN 76312087 Ki = 71.5 nM T07806 C3A8EB 76312089 Ki = 911.6 nM T07806 COM84H 76315630 Ki = 2478 nM T07806 CR0XQ1 76319309 Ki = 2317 nM T07806 CU6YO0 76322954 Ki = 36.4 nM T07806 CP3YB5 76322955 Ki = 6692 nM T07806 C3IPW2 76322957 Ki = 751.8 nM T07806 CDY2S1 76326510 Ki = 1249 nM T07806 C6LUP2 76326511 Ki = 1456 nM T07806 C2Z5SX 76326513 Ki > 10000 nM T07806 CNU59S 76326515 Ki = 833 nM T07806 C5HJ9N 76330154 Ki = 2748 nM T07806 C1XTC0 76330155 Ki = 3641 nM T07806 C9SX2Q 76330156 Ki = 4197 nM T07806 C70ZVB 86221574 Ki = 7596 nM T07806 CEMZ15 118464420 Ki > 10000 nM T07806 CV2L6O 118464425 Ki = 9653 nM T07806 CFNG86 118464427 Ki > 10000 nM T07806 C7AYV5 118540795 EC50 > 10000 nM T07806 C5X8MN 122186880 IC50 = 1000 nM T07806 CJ26IS 122187375 Ki = 1608 nM T07806 C7RP0M 122187378 Ki = 2466 nM T07806 C7ODW3 122195524 Ki > 900 nM T07806 C3VDY7 122197403 Ki = 114 nM T07806 C1MFJ3 122197404 Ki > 1000 nM T07806 C7GO0U 122197405 Ki = 88 nM T07806 CO63ET 122483280 Ki = 3744 nM T07806 C4QM2E 124247485 Ki > 10000 nM T07806 CTBN56 127026052 Ki = 1778.28 nM T07806 CBE56W 127026514 Ki = 845 nM T07806 CZ61LK 127034966 IC50 > 5011.87 nM T07806 CA0SN5 127034967 EC50 > 5011.87 nM T07806 CU49VE 127036186 Ki = 1348.96 nM T07806 CG06BD 127036932 Ki = 891.25 nM T07806 CVW71O 127036953 Ki = 954.99 nM T07806 C50GOC 130442480 Ki = 8800 nM T07806 CM04RF 130442572 Ki = 9300 nM T07806 CY8B9L 132060743 Ki = 1431 nM T07806 CGHO19 132060770 Ki = 2438 nM T07806 CAVB41 132584404 Ki > 10000 nM T07806 CBU81N 134149168 Ki > 10000 nM T07806 C1GY2T 135156251 EC50 > 10000 nM T07806 C6N8GM 135367405 Ki > 10000 nM T07806 C6LU0C 135367816 Ki > 10000 nM T07806 CD2TH9 135367820 Ki > 10000 nM T07806 C5AMD9 135367857 Ki > 10000 nM T07806 CUKO20 136020617 Ki > 10000 nM T07806 COF0U5 136020618 Ki > 10 nM T07806 CF89JI 136030596 Ki > 10000 nM T07806 CE8GB9 136030693 Ki > 10000 nM T07806 C65VFI 136030744 Ki > 10000 nM T07806 COIX80 136054961 Ki > 10000 nM T07806 CS0JL5 136118616 Ki > 10000 nM T07806 C5UDW3 136118620 Ki > 10000 nM T07806 C8I6UN 136118621 Ki > 10000 nM T07806 CD7OE2 136118652 Ki > 10000 nM T07806 C42FCS 136118661 Ki > 10000 nM T07806 CAE39V 136188797 Ki > 10000 nM T07806 CLAP52 136259032 Ki > 10000 nM T07806 C8RYA2 137634921 EC50 = 570 nM T07806 CPI68E 137646281 Ki = 2032 nM T07806 CHDN35 145964150 EC50 = 29 nM T07806 C12OVL 145965034 Ki > 10000 nM T07806 C5W4LM 145965940 Ki > 10000 nM T07806 C81VUO 145967771 Ki > 10 nM T07806 CJS56K 145967795 Ki > 10000 nM T07806 CQJ5O8 145971635 Ki > 10000 nM T07806 C79TNE 145972796 Ki > 10000 nM T07806 C6XIN0 145974114 Ki > 10000 nM T07806 CD8ZL6 145974750 Ki > 10 nM T07806 C71CYU 145975946 EC50 = 180 nM T07806 C6BFY7 145977338 Ki > 10000 nM T07806 C3BI1R 145978113 Ki > 10000 nM T07806 CQU8R0 145978665 Ki > 10000 nM T07806 C6AV9G 145978819 Ki > 10000 nM T07806 C86XQR 145988313 Ki = 3406 nM T07806 C4GV8Q 145990586 Ki = 1209 nM T07806 CC2G1V 146025727 Ki = 9900 nM T07806 C6P3SR 153287553 Ki > 10000 nM T07806 CV9G7Z 153287572 Ki > 10000 nM T07806 CO85KL 153287574 Ki > 10000 nM T07806 CUSA24 155519891 Ki > 10000 nM T07806 CB79ZW 155536080 Ki > 10000 nM T07806 C3N9VU 10251906 Ki > 500 nM T07806 D00FHZ 124007 EC50 > 10000 nM T07806 D01HRV 9847194 IC50 = 150 nM T07806 D01KAX 135453290 Ki > 10000 nM T07806 D02EPZ 24782016 Ki > 10000 nM T07806 D02NNS 9845181 Ki = 7700 nM T07806 D02UWB 1809 Ki = 1.259 nM T07806 D03DET 10287730 Ki = 199.53 nM T07806 D03JOX 11311147 IC50 > 10000 nM T07806 D03KPA 15870567 Ki = 1625 nM T07806 D03MVY 10198700 Ki = 32 nM T07806 D03TDN 1342 Ki = 10.1 nM T07806 D03XAE 10775128 Ki = 5.5 nM T07806 D04AQE 1833 Ki = 3.5 nM T07806 D04DLR 128018 Ki = 12.1 nM T07806 D05GDP 599482 Ki > 10000 nM T07806 D05XGR 6918647 Ki = 398.11 nM T07806 D05ZUX 44207909 Ki >= 1000 nM T07806 D06QGD 11357862 IC50 > 10000 nM T07806 D07LRJ 5312149 Ki = 794.33 nM T07806 D07ZOP 11470616 IC50 > 10000 nM T07806 D08CKM 9863250 Ki = 1584.89 nM T07806 D09AVG 11831220 Ki = 353 nM T07806 D09HJL 10331436 Ki = 3300 nM T07806 D09OYA 2107 Ki = 250 nM T07806 D09PIN 3378093 Ki = 6.31 nM T07806 D09RPR 16737207 Ki > 10000 nM T07806 D09WIL 10028436 Ki = 630.96 nM T07806 D0C3EX 1797 Ki = 1.2 nM T07806 D0C5XQ 1832 IC50 = 550 nM T07806 D0D8GV 9830741 Ki > 500 nM T07806 D0D9YW 3292447 Ki = 1 nM T07806 D0F0IA 11301655 Ki > 2000 nM T07806 D0F6CD 5202 Ki = 1.1 nM T07806 D0FF6S 16038374 IC50 > 10000 nM T07806 D0G7QT 10131112 IC50 = 110 nM T07806 D0H7PC 6918553 Ki > 3981.07 nM T07806 D0H9QG 5312148 Ki < 5011.87 nM T07806 D0I9KV 11220599 IC50 > 10000 nM T07806 D0K9MT 10912152 Ki = 472 nM T07806 D0KQ9H 10468938 IC50 = 28 nM T07806 D0KS0I 24894910 EC50 > 10000 nM T07806 D0L5MW 181743 Ki = 100 nM T07806 D0M7SY 9910352 Ki = 630.96 nM T07806 D0O3GF 1220 EC50 = 260 nM T07806 D0PN8D 44351692 Ki = 2 nM T07806 D0QM3E 9870500 Ki = 3.981 nM T07806 D0R3GW 10296414 Ki = 10 nM T07806 D0T2RY 9948320 Ki >= 1000 nM T07806 D0V7OO 10386282 IC50 = 47 nM T07806 D0X8LG 11243002 IC50 > 10000 nM T08298 CJGI52 44309728 Ki = 13 nM T08298 CV7O8U 44309729 Ki = 16 nM T08298 C1IY3Z 44309748 Ki = 38 nM T08298 C9RLK1 44309811 Ki = 8 nM T08298 CRP69J 44309881 Ki = 270 nM T08298 CJQ3D0 44309888 Ki = 133 nM T08298 C5GB2O 44309904 Ki = 122 nM T08298 CRJ58I 44309905 Ki = 13 nM T08298 CZ1Q0D 44309956 Ki = 2300 nM T08298 C2VW1E 44309957 Ki = 85 nM T08298 CFRP17 44310015 Ki = 75 nM T08298 CGNM89 44310088 Ki = 74 nM T08298 CL46EF 44310108 Ki = 360 nM T08298 C0U5VJ 44310111 Ki = 580 nM T08298 CX31HT 44310132 Ki = 80 nM T08298 CYD20K 44310147 Ki = 7 nM T08298 CAY7G2 44453610 Ki = 8 nM T08298 CF9UM2 44453613 Ki = 7 nM T08298 CS6NG3 44453636 Ki = 85 nM T08298 C78DJQ 71711730 IC50 < 10000 nM T08298 CDQ62V 137637214 Ki > 50000 nM T08298 C2K8JV 137639385 Ki > 50000 nM T08298 CNX46H 137654508 Ki > 50000 nM T08298 D0Y7HC 44310146 Ki = 7 nM T76685 D07ILQ 4671 Ki > 5000 nM T76685 D0E6YQ 1935 Ki > 1000 nM T76685 D0L7AS 5284592 Ki = 2.19 nM T76685 D0O1UZ 644019 Ki = 1459 nM T76685 D0O3OS 104850 EC50 = 0.11 nM T76685 D0P1FO 16078 Ki = 2.9 nM T76685 D0R1RS 3715 Ki > 20000 nM T76685 D0T9TJ 3034010 IC50 <= 100 nM T76685 D0U5CE 1548943 Ki > 10000 nM T76685 D08DGC 3083542 Ki = 5.7 nM T76685 D0I4PW 60164925 EC50 > 10000 nM T76685 D0J6KZ 57331749 IC50 > 2000 nM T76685 D0LI1C 44469321 IC50 > 10000 nM T76685 D0P5CM 56945146 IC50 = 5000 nM T76685 D0Q7NB 10253143 EC50 > 10000 nM T76685 D0Q8WG 67029278 EC50 = 854 nM T76685 D0U2BH 65064 Ki = 33600 nM T76685 D0VH3H 49779607 Ki = 3 nM T76685 D0W3GL 9849616 Ki = 3.5 nM T76685 D0Y9RO 107778 EC50 = 0.6 nM T76685 D00GES 66553204 IC50 = 0.5 nM T76685 D00BXK 25027058 IC50 = 1.5 nM T76685 D01RIT 24857045 IC50 = 21.6 nM T76685 D02ZVY 72712999 Ki = 3.57 nM T76685 D04ZLC 66547077 IC50 = 400 nM T76685 D05GDS 66547073 IC50 = 1 nM T76685 D07BFP 60148509 Ki = 324 nM T76685 D07IHT 4296438 Ki > 20000 nM T76685 D07NAA 24945235 EC50 = 1 nM T76685 D0D1EI 72713196 Ki = 19.47 nM T76685 D0DE0C 72713199 Ki = 1.54 nM T76685 D0E6YT 71539748 Ki > 60000 nM T76685 D0FR1Q 13458368 EC50 > 10000 nM T76685 D0FS0D 44571565 EC50 = 50.7 nM T76685 D0GQ8W 46871948 EC50 = 118.3 nM T76685 D0GX6V 23624319 Ki = 13 nM T76685 D0I1XE 72713197 Ki = 1.93 nM T76685 D0J5XM 25098114 IC50 = 11 nM T76685 D0KX2W 46889224 Ki = 8.9 nM T76685 D0M2RT 24863732 Ki = 20 nM T76685 D0O4RN 24744027 EC50 = 1 nM T76685 D0S3RX 44571486 IC50 = 1173.2 nM T76685 D0TI3Q 11555526 Ki = 11.9 nM T76685 D0V0UW 25098092 IC50 = 1.9 nM T76685 D0WJ3F 71584280 Ki = 1297 nM T76685 D0WK8I 44582884 EC50 = 300 nM T76685 D0YZ8I 4273754 Ki = 383 nM T76685 D0Z8WF 24944528 IC50 = 1 nM T76685 D03ACT 9844711 Ki >= 10000 nM T76685 D06TGE 11226090 IC50 = 0.29 nM T76685 D0A9OR 11179267 IC50 = 1.905 nM T76685 D0H1FL 11316919 Ki = 0.82 nM T76685 D0J0AE 10052040 Ki = 0.12 nM T76685 D0J7RW 5311501 Ki = 1.89 nM T76685 C1S7VI 2415 Ki > 20000 nM T76685 C5H9CN 9287 Ki > 10000 nM T76685 CQP80E 15339 Ki > 20000 nM T76685 C9WJ7H 25957 Ki > 10000 nM T76685 C3ERF2 30219 Ki = 714 nM T76685 CWYV98 39860 Ki = 3.981 nM T76685 CTK25Q 72277 Ki = 35700 nM T76685 C8SD5O 72300 Ki = 3150 nM T76685 C0AGE7 78262 Ki > 10000 nM T76685 CJ5T2N 98523 Ki = 24 nM T76685 C0QSW4 104849 Ki = 5.4 nM T76685 CNIW58 107905 Ki = 47300 nM T76685 CR4JB5 129128 Ki = 23 nM T76685 CRYZ13 169652 Ki = 65 nM T76685 CMP4K1 192007 Ki = 5668 nM T76685 C4P1GV 194130 Ki = 38.8 nM T76685 C3T5KU 292955 Ki > 10000 nM T76685 CVL1A0 320263 Ki = 21100 nM T76685 CL3UD5 320264 Ki > 10000 nM T76685 C94GYM 331257 EC50 > 10000 nM T76685 CFY02L 356017 Ki > 10000 nM T76685 C8X7ST 356018 Ki > 10000 nM T76685 C5V0SH 386338 Ki = 1200 nM T76685 C8LY2I 391240 Ki > 10000 nM T76685 CJ3NQ1 601368 IC50 > 10000 nM T76685 CU57BO 601392 IC50 > 10000 nM T76685 C37RCW 622545 EC50 = 565 nM T76685 CPK8U9 695120 Ki > 10000 nM T76685 CZ9SJ1 695133 Ki > 10000 nM T76685 CECS97 708647 Ki = 1288 nM T76685 CGT6F3 738959 Ki > 10000 nM T76685 CS0P7U 743023 EC50 < 10000 nM T76685 CMR9E1 746182 Ki > 10000 nM T76685 CT7DE5 759445 Ki = 1000 nM T76685 C3VXW6 836750 Ki > 10000 nM T76685 CDE0L5 853260 EC50 > 100000 nM T76685 C90NZF 853261 EC50 = 2600 nM T76685 CV24TH 868829 Ki > 10000 nM T76685 CVRG42 872331 Ki > 10000 nM T76685 CQ3K8M 897320 Ki > 10000 nM T76685 C7SQL6 900707 Ki > 10000 nM T76685 COU5J2 900710 Ki > 10000 nM T76685 C6D7XU 991033 Ki > 20000 nM T76685 C1L2CV 1000896 Ki > 50 nM T76685 C6SDA3 1001644 Ki = 1600 nM T76685 CB79QJ 1034762 Ki = 1373.03 nM T76685 CTXK08 1040500 Ki > 10000 nM T76685 CT1W9S 1043357 IC50 = 50.12 nM T76685 CFY2M3 1075977 Ki = 106 nM T76685 C12KOP 1087788 IC50 = 199.53 nM T76685 C8PEU1 1087790 IC50 = 39.81 nM T76685 CN6D0T 1089375 EC50 < 10000 nM T76685 CZR2G8 1098594 Ki > 10000 nM T76685 CCE93A 1101768 IC50 = 1.259 nM T76685 CZJA94 1107142 EC50 = 50.12 nM T76685 C4LD2S 1117960 EC50 = 630.96 nM T76685 C06QRH 1124158 IC50 < 10000 nM T76685 C0AGV1 1124172 IC50 = 31.62 nM T76685 C4NL1G 1127069 Ki = 1100 nM T76685 C98QPF 1130139 IC50 = 290 nM T76685 C1GSP2 1144102 EC50 < 10000 nM T76685 C8O0RS 1202067 IC50 = 4543 nM T76685 C0MYU2 1281700 Ki > 10000 nM T76685 C8KD9F 1281702 Ki > 10000 nM T76685 CH8PY0 1281704 Ki > 10000 nM T76685 CX5F6G 1281706 Ki > 10000 nM T76685 CPMN31 1315417 EC50 = 63.1 nM T76685 CM2D5Q 1350471 EC50 = 251 nM T76685 C9EMW7 1548023 EC50 < 10000 nM T76685 C7UPS9 1602258 Ki > 50 nM T76685 C3CZ0N 1626958 EC50 = 630.96 nM T76685 CF57VU 1649385 Ki > 10000 nM T76685 CZ71FX 1722112 Ki > 10000 nM T76685 CT42LA 1837112 Ki > 50 nM T76685 CYT1G7 2057275 EC50 < 10000 nM T76685 C6F1EP 2084332 EC50 > 100000 nM T76685 CC0Y2N 2086721 EC50 = 5910 nM T76685 C3WIV0 2117799 Ki = 800 nM T76685 CM4S0X 2188265 Ki > 50 nM T76685 C5B6FD 2317892 EC50 = 390 nM T76685 CIT03M 2323038 Ki > 10000 nM T76685 CWJ02B 2334657 IC50 = 1258.93 nM T76685 C62SYO 2691386 EC50 = 314.1 nM T76685 C4IGL3 2729560 IC50 = 4200 nM T76685 C95VEI 2729564 EC50 = 1 nM T76685 C9NS7Q 2740778 EC50 > 10000 nM T76685 CO04GZ 2787166 EC50 > 10000 nM T76685 CIUG12 2787170 EC50 > 10000 nM T76685 CYG2A9 2801231 EC50 = 420 nM T76685 CU0JC7 2814417 Ki = 1606 nM T76685 C85HRJ 2836420 Ki = 272 nM T76685 CSEB28 2836426 EC50 > 10000 nM T76685 CDTK31 2846758 Ki = 1008.48 nM T76685 C7SD1X 2850042 Ki > 10000 nM T76685 C9JT7I 2851184 EC50 > 10000 nM T76685 C9HCD2 2853642 Ki = 185.14 nM T76685 CI04TU 2987572 EC50 > 10000 nM T76685 CW1QZ9 3145647 Ki = 2314 nM T76685 CF0B1H 3154042 Ki = 2785 nM T76685 CX9Z5T 3158002 EC50 = 630.96 nM T76685 C5MKT8 3168799 Ki > 50 nM T76685 C8KH0Z 3258886 Ki > 10000 nM T76685 CE24BQ 3298404 Ki > 10000 nM T76685 CQ38BO 3340785 Ki = 193 nM T76685 CLCV10 3372949 Ki = 1530 nM T76685 CSU8B7 3379236 Ki = 108 nM T76685 CCQZ29 3426415 Ki = 264 nM T76685 C2C9PX 3579176 EC50 > 10000 nM T76685 C29OCP 3604821 IC50 = 5011.87 nM T76685 C08PSA 3643741 Ki > 10000 nM T76685 CTS89I 3703767 Ki = 325 nM T76685 CVBD75 3717285 Ki = 1177 nM T76685 CTEP25 3746369 Ki = 2716 nM T76685 C2PJ9B 3840634 Ki = 273 nM T76685 CA1O6R 3868445 EC50 = 0.6 nM T76685 C8O1VI 3929482 IC50 = 0.7943 nM T76685 CJ2D3A 3932001 EC50 = 200 nM T76685 CIJ95Y 4055807 Ki = 92 nM T76685 C5OVS7 4140053 EC50 > 10000 nM T76685 CQD4C6 4164761 EC50 = 440 nM T76685 CEO84R 4195510 Ki = 520 nM T76685 C9SG4D 4239464 Ki = 875 nM T76685 CM31EP 4262768 EC50 = 895.6 nM T76685 C17EFM 4297602 Ki = 7490 nM T76685 C6K2SR 4346308 Ki = 520 nM T76685 C1EJ3I 4399268 Ki = 2593 nM T76685 CEM60H 4402318 EC50 = 8.1 nM T76685 C5IJ2F 4458788 EC50 > 10000 nM T76685 C7ROQ6 4544649 Ki = 1764 nM T76685 CXC9U2 4554609 Ki > 10000 nM T76685 CBC0D2 4559116 Ki > 10000 nM T76685 C5PA1K 4621779 Ki = 94 nM T76685 CG6T9V 4677403 Ki = 3949 nM T76685 C13HIO 4693083 IC50 = 1584.89 nM T76685 CUCD57 4693614 EC50 = 200 nM T76685 CO0EK1 4736636 Ki = 227 nM T76685 C64KTC 4807210 IC50 = 3500 nM T76685 CFK3L2 4831482 IC50 = 1584.89 nM T76685 C95ORJ 4877853 IC50 = 398.11 nM T76685 CDT56R 4880561 IC50 = 1995.26 nM T76685 C56SGI 4963989 Ki = 82 nM T76685 C0LK2Z 4996150 Ki = 308 nM T76685 C83IAN 5019347 EC50 > 10000 nM T76685 CET70S 5031403 Ki = 1030 nM T76685 C8YKU2 5042131 Ki = 1943 nM T76685 CX46YD 5164405 Ki > 10000 nM T76685 C0FI8Q 5283393 Ki = 9600 nM T76685 CG7MQ8 5283394 Ki = 7.3 nM T76685 C2O5ZR 5283396 Ki = 30 nM T76685 CCY68Q 5283399 Ki = 1860 nM T76685 C4SM0G 5283403 Ki = 13 nM T76685 C2KND4 5283410 Ki = 4980 nM T76685 C0VUE9 5283444 Ki > 1500 nM T76685 CCM3H2 5283452 Ki > 10000 nM T76685 CY7ZM6 5283455 Ki = 53 nM T76685 CJ5I8L 5283456 Ki = 41 nM T76685 C3J9NW 5285645 EC50 > 30000 nM T76685 CZ46HG 5315659 Ki = 760 nM T76685 CK0X9M 5318518 IC50 = 100 nM T76685 C47FZC 5319201 Ki > 10000 nM T76685 CIU1J6 5321844 IC50 = 4600 nM T76685 CJI57N 5321851 Ki = 2260 nM T76685 CP9GM8 5322490 Ki = 2396 nM T76685 CPFC04 5368482 Ki > 40000 nM T76685 CZ31XM 5722610 IC50 > 50000 nM T76685 C8EB7Q 5854591 Ki = 1000 nM T76685 CC4B0K 5917569 Ki > 10000 nM T76685 C0JQ4U 6401059 EC50 > 30000 nM T76685 C8FQ6P 6413892 Ki = 2269 nM T76685 C3RNJ8 6434324 IC50 = 15200 nM T76685 CWF02M 6440803 Ki > 10000 nM T76685 CF2B7X 6442405 Ki > 20000 nM T76685 C4WPT9 6453891 Ki = 15 nM T76685 C3TLF8 6481606 Ki > 10000 nM T76685 CPLC65 6481633 Ki > 10000 nM T76685 C2C4KE 6604176 Ki = 9.2 nM T76685 CP6RW5 6621153 Ki = 5 nM T76685 C1ZW6X 6973727 IC50 > 17000 nM T76685 CRWD27 7620138 Ki = 560 nM T76685 CDUC94 7620149 Ki = 960 nM T76685 CO3M5A 7620714 Ki = 56 nM T76685 C16AMB 7620725 Ki = 9.6 nM T76685 CGP17E 7921574 EC50 = 90 nM T76685 C7H2FT 7929121 Ki = 1100 nM T76685 C45OEP 8178387 Ki = 33 nM T76685 CPM3X1 8712703 Ki = 260 nM T76685 CL3DG9 8916493 EC50 > 30000 nM T76685 C8E0JX 8916569 EC50 > 30000 nM T76685 C7I8PY 9123860 Ki > 10000 nM T76685 CGFY81 9123866 Ki > 10000 nM T76685 CQ3S9L 9124038 Ki > 10000 nM T76685 CZLT78 9192580 Ki > 10000 nM T76685 C32SMR 9401432 Ki > 10000 nM T76685 CH0V2X 9456049 Ki > 10000 nM T76685 CVZG73 9799417 EC50 = 6.1 nM T76685 CTA5Z1 9800032 Ki = 908 nM T76685 C9V2CG 9800960 Ki = 2.43 nM T76685 C0CQX1 9810861 Ki < 100 nM T76685 CWGT52 9825614 Ki = 4315 nM T76685 CVR42O 9826744 Ki = 0.42 nM T76685 CUL5C1 9828471 IC50 = 94 nM T76685 CU96OX 9829238 Ki = 4 nM T76685 COD3T8 9829239 Ki = 8.4 nM T76685 C94AQK 9840457 IC50 = 79 nM T76685 CRM5P4 9845561 Ki = 0.46 nM T76685 CJLR93 9847217 IC50 = 4 nM T76685 CQWX41 9867382 Ki = 1.86 nM T76685 C9Q2UN 9867770 Ki = 2370 nM T76685 CRP37G 9868656 IC50 = 2.5 nM T76685 C1RO9M 9887568 Ki = 7050 nM T76685 CJG8R5 9888694 Ki > 10000 nM T76685 C6JD8A 9906800 IC50 = 766 nM T76685 CGP96L 9909689 Ki = 0.86 nM T76685 CB4L7I 9911463 Ki = 1917 nM T76685 C95PSM 9912393 Ki > 1000 nM T76685 CT4GD0 9914194 Ki > 1000 nM T76685 CU67PO 9933988 IC50 = 56 nM T76685 CF92JW 9935463 IC50 = 3.5 nM T76685 CLU0R5 9949177 Ki = 2.7 nM T76685 CI8F4E 9952038 Ki = 877 nM T76685 C7BXH9 9956047 Ki = 16 nM T76685 CXF43E 9956414 Ki = 23000 nM T76685 CZ7DT6 9968042 IC50 = 19000 nM T76685 CLD4O3 9968810 IC50 = 1800 nM T76685 C5SRP1 9971539 Ki = 87 nM T76685 C9LYH8 9975456 Ki = 0.34 nM T76685 C07RPH 9976253 Ki = 2.72 nM T76685 C5B0KC 10002952 Ki = 0.32 nM T76685 C6PFI7 10006706 Ki = 2.9 nM T76685 CIJ08V 10008091 Ki = 1.1 nM T76685 CNI7K3 10024106 EC50 = 1.2 nM T76685 C2EK3Y 10024236 Ki = 15 nM T76685 C3MN1Y 10028104 Ki = 308 nM T76685 CXQ29Y 10028229 IC50 = 5.4 nM T76685 CA06TQ 10028888 IC50 = 4.3 nM T76685 C6EML8 10029316 IC50 = 0.39 nM T76685 C8MLU5 10029650 Ki = 8.9 nM T76685 C76EVS 10031352 Ki = 1.4 nM T76685 CJT1O5 10045570 Ki = 82 nM T76685 CUJV52 10045631 Ki = 28 nM T76685 CM7B9Q 10052826 IC50 = 4.3 nM T76685 CX53LI 10053649 Ki = 204 nM T76685 C29SQA 10073313 EC50 > 3162.28 nM T76685 C09GTF 10076710 Ki = 3.6 nM T76685 CX1R2V 10077379 Ki = 5.8 nM T76685 CB34HN 10084135 IC50 = 7400 nM T76685 C6CB0K 10091328 Ki = 22.3 nM T76685 CFY07G 10091392 EC50 = 25.12 nM T76685 C3SGD4 10091426 Ki = 1000 nM T76685 CZ5F8M 10094322 EC50 > 3162.28 nM T76685 C0X3PA 10097077 Ki = 5 nM T76685 CETX82 10097960 Ki = 13 nM T76685 CF2ZS1 10099858 Ki = 2 nM T76685 C3KG5H 10109902 IC50 = 3467.37 nM T76685 CQ7C4M 10112443 IC50 = 1500 nM T76685 C5TH1Q 10112572 Ki = 29 nM T76685 C27MKW 10114327 Ki = 14 nM T76685 CJ81FH 10116471 IC50 = 8 nM T76685 CHW60K 10126513 IC50 = 6 nM T76685 C2ZKH6 10127040 IC50 = 80 nM T76685 C2W7ET 10127144 IC50 = 12 nM T76685 C6X9EY 10127451 IC50 = 53 nM T76685 CRZ04L 10127496 Ki = 33 nM T76685 CRML57 10127677 IC50 = 480 nM T76685 CYJ69P 10127751 IC50 = 1.9 nM T76685 C60BYH 10127897 IC50 = 35 nM T76685 CRI8P0 10128697 IC50 = 1.3 nM T76685 CSW06O 10134835 IC50 = 900 nM T76685 C9XQ1F 10136173 IC50 = 631 nM T76685 CO9KZ4 10140173 Ki = 5.7 nM T76685 C4VC9R 10141881 Ki = 3.7 nM T76685 CG1RJ0 10151599 IC50 = 210 nM T76685 CVO6Z3 10151737 IC50 = 10 nM T76685 CM4D1E 10151772 IC50 = 17 nM T76685 CPEK39 10151837 IC50 = 31 nM T76685 C3Q9WV 10151871 IC50 = 11 nM T76685 CFI4R1 10152346 IC50 = 5.7 nM T76685 C7SAR0 10152529 IC50 = 0.302 nM T76685 C0SK2N 10152740 IC50 = 5.2 nM T76685 C0O2NM 10153212 Ki = 4100 nM T76685 C78NUA 10155451 IC50 = 1900 nM T76685 CD48QZ 10157119 IC50 = 467.74 nM T76685 CVH78W 10157922 IC50 = 900 nM T76685 CPAX61 10159759 Ki = 29 nM T76685 CZ3E4L 10173396 IC50 = 16.6 nM T76685 CR9PF2 10173886 IC50 = 95 nM T76685 C42WGZ 10174045 Ki = 334 nM T76685 CLP8Z2 10174286 IC50 = 3.7 nM T76685 CB7SK3 10174641 IC50 = 1 nM T76685 CGV5Z1 10174842 IC50 = 3.1 nM T76685 CL40OZ 10182828 IC50 = 60 nM T76685 CY8J0G 10183243 IC50 = 190 nM T76685 C2QE6Z 10186399 Ki = 5.8 nM T76685 C7GIW8 10194245 IC50 = 2800 nM T76685 CV9HS6 10194582 IC50 = 21 nM T76685 CY4EQ6 10195058 IC50 = 11 nM T76685 CS49KR 10195276 IC50 = 29 nM T76685 CRDN48 10195347 Ki = 35 nM T76685 CS1V9E 10195397 Ki = 197 nM T76685 CS2O5P 10195715 IC50 = 4 nM T76685 CY4O5A 10195774 IC50 = 20 nM T76685 C6XY7L 10196577 IC50 = 1.8 nM T76685 C5UFP0 10200053 Ki = 97 nM T76685 CQU58G 10202808 EC50 = 500 nM T76685 C23ZAH 10202883 EC50 = 100 nM T76685 CD5RA2 10203016 IC50 = 3100 nM T76685 C9HNG7 10204999 IC50 = 46 nM T76685 C3PSB2 10205057 EC50 = 5 nM T76685 COX02C 10207068 IC50 = 16 nM T76685 CCF80H 10216046 Ki = 122 nM T76685 CZBY62 10216322 IC50 = 119 nM T76685 CK4I2M 10216436 IC50 = 8 nM T76685 CX6R8Y 10216582 IC50 = 1578 nM T76685 CF5QE0 10216596 IC50 = 4 nM T76685 C41QVC 10216983 IC50 = 32 nM T76685 CD3M8S 10216984 Ki = 27 nM T76685 CTK1E8 10217134 IC50 = 210 nM T76685 CK1NV9 10217165 IC50 = 14 nM T76685 CF02BR 10217166 IC50 = 65 nM T76685 CRW69G 10217167 IC50 = 43 nM T76685 CY6G4H 10217386 IC50 = 32 nM T76685 CHOI31 10217488 IC50 = 6.3 nM T76685 CM3Z2D 10217960 IC50 = 11 nM T76685 CGD2O6 10218033 IC50 = 3.9 nM T76685 CQ45ZC 10218471 IC50 = 1.5 nM T76685 CDF3J9 10220912 IC50 = 9 nM T76685 CZH07C 10227475 IC50 = 70 nM T76685 C51GDE 10227614 Ki = 4000 nM T76685 CUI75O 10236980 IC50 = 5623.41 nM T76685 CQ35RS 10238098 IC50 = 174 nM T76685 CWK23N 10239221 IC50 = 3.4 nM T76685 CL3C6O 10250275 Ki = 638 nM T76685 CB04DY 10250276 Ki = 20 nM T76685 C5RHE4 10252734 Ki = 363 nM T76685 CUF43P 10254284 IC50 = 5.5 nM T76685 C7ZMF9 10254993 Ki = 4 nM T76685 CU6S3K 10257361 Ki = 10 nM T76685 CQRW06 10273200 IC50 = 1100 nM T76685 C85OJI 10275599 IC50 = 17 nM T76685 CX25NI 10276190 Ki = 5 nM T76685 C96ABX 10276669 IC50 = 169.82 nM T76685 CWU0X7 10277271 IC50 = 4.1 nM T76685 CX4TI3 10278467 IC50 = 5.2 nM T76685 CM86TS 10287827 IC50 = 10 nM T76685 CL2E0G 10288440 IC50 = 1.514 nM T76685 CHYX37 10288473 IC50 = 1.122 nM T76685 CB64KF 10289044 IC50 = 21 nM T76685 C1RBL0 10289123 IC50 = 5.8 nM T76685 CU45SK 10294778 Ki > 5000 nM T76685 C1Y0XC 10295316 IC50 = 6000 nM T76685 C3KJ2P 10296307 IC50 = 540 nM T76685 CQR29X 10297613 Ki = 23 nM T76685 CIXD91 10309464 IC50 = 13 nM T76685 C3M9SA 10310004 IC50 = 763 nM T76685 CX4U9T 10310427 IC50 = 340 nM T76685 COE0K9 10310644 IC50 = 6.6 nM T76685 C35JNY 10310812 IC50 = 14 nM T76685 CG3M2Y 10310945 IC50 = 5.7 nM T76685 C78QAR 10311022 IC50 = 26 nM T76685 CE4HG6 10311095 IC50 = 154 nM T76685 C08NME 10311098 IC50 = 7 nM T76685 CU34MP 10311368 IC50 = 2.9 nM T76685 CRP35L 10311846 IC50 = 1.9 nM T76685 CHOT95 10312127 Ki > 5000 nM T76685 C27TCH 10319351 Ki = 2.512 nM T76685 C5PXW2 10319620 Ki = 88 nM T76685 CI20DM 10324989 Ki = 905 nM T76685 COU9I0 10340138 Ki = 0.73 nM T76685 CPNT75 10342137 Ki = 38 nM T76685 CJKP36 10346150 Ki = 97.9 nM T76685 C6F7DJ 10346347 Ki = 4534 nM T76685 C2G8IR 10346644 Ki = 0.1 nM T76685 C1J7HS 10349119 Ki = 5 nM T76685 C7SW3C 10360860 Ki = 9.5 nM T76685 CDR50J 10361702 Ki = 0.4365 nM T76685 CI2MZ3 10366006 IC50 = 20 nM T76685 CJHV10 10366839 IC50 = 1.318 nM T76685 CLVC49 10367110 Ki = 1.8 nM T76685 C5QT1A 10367921 IC50 = 0.58 nM T76685 COFR51 10368712 Ki = 9 nM T76685 C73FXG 10369017 Ki = 178 nM T76685 CH4M5K 10370677 Ki > 10000 nM T76685 CD6MC9 10382701 Ki = 1.995 nM T76685 C7HV9R 10383130 Ki = 297 nM T76685 CJ4NL2 10385575 EC50 > 3162.28 nM T76685 CIK8N3 10386267 Ki = 2838 nM T76685 CQ3M6K 10391336 Ki = 2 nM T76685 C94LNA 10407148 Ki = 7.42 nM T76685 CM1C5I 10407577 Ki = 0.94 nM T76685 C9Y3TJ 10410512 IC50 = 56 nM T76685 CHK4R7 10413523 IC50 = 1.2 nM T76685 C2BT6D 10413635 Ki = 62.95 nM T76685 CLFB89 10413921 Ki = 76.7 nM T76685 CI39ZO 10433670 IC50 = 17 nM T76685 CO1GI7 10435654 Ki = 0.00035 nM T76685 C36LVH 10438646 Ki = 4.9 nM T76685 CFWR83 10449945 Ki = 79.1 nM T76685 C5OGQ1 10452791 Ki = 50 nM T76685 CA9EN5 10453633 Ki = 0.5 nM T76685 C97LHV 10454092 EC50 > 30 nM T76685 C2JX0C 10456931 IC50 = 1.9 nM T76685 CPJ38R 10461516 Ki = 2.5 nM T76685 CWU17B 10461605 Ki = 2.5 nM T76685 C73TBN 10468802 Ki > 10000 nM T76685 CV1S8R 10478331 IC50 = 4.3 nM T76685 CCEA61 10479060 Ki = 48.3 nM T76685 CW0K3P 10479686 Ki = 227 nM T76685 C93ZIS 10479729 Ki = 103.2 nM T76685 CXFJ90 10482705 Ki = 25 nM T76685 CU68XN 10483071 Ki = 1.3 nM T76685 CY5Q3L 10500128 Ki = 0.1 nM T76685 CY1Z0O 10500863 Ki = 558 nM T76685 C3HE0R 10522112 Ki = 2.17 nM T76685 CH1NY0 10527931 Ki = 1.5 nM T76685 C1NS8A 10531071 Ki = 29 nM T76685 CLZ9Q7 10545949 Ki > 10000 nM T76685 CZ67QE 10546891 Ki = 2 nM T76685 C2YTM0 10546947 Ki = 148 nM T76685 C0N3JX 10548081 IC50 = 7000 nM T76685 CN6CJ9 10566956 Ki = 875 nM T76685 CB8L6S 10577158 Ki > 10000 nM T76685 C4WX2N 10596625 Ki > 10000 nM T76685 CEF0Y9 10597702 Ki = 14 nM T76685 C7Q6NW 10618930 Ki = 1 nM T76685 CLE3D5 10619854 Ki = 2.84 nM T76685 CQG23I 10639725 Ki = 42 nM T76685 CP07NE 10642025 Ki = 21.7 nM T76685 CSG1E4 10646233 Ki = 122.7 nM T76685 CNE1B0 10647307 Ki > 10000 nM T76685 C34ADC 10650400 Ki = 60 nM T76685 C40THY 10667130 Ki = 700 nM T76685 CLU8K3 10667559 Ki = 1945 nM T76685 CE5I1M 10672879 Ki = 187 nM T76685 CN0IJ1 10673015 Ki > 10000 nM T76685 C9JFU2 10673782 Ki = 18 nM T76685 C6C4KH 10687450 Ki = 204 nM T76685 C2JR1N 10694463 Ki = 13 nM T76685 C1W3QS 10713019 Ki = 33 nM T76685 C4D5LN 10717065 Ki = 0.43 nM T76685 CE8Q6I 10720372 Ki > 20000 nM T76685 CDNT67 10721387 Ki > 10000 nM T76685 CHN83D 10738579 Ki = 681 nM T76685 CZLI34 10742513 Ki = 9.2 nM T76685 C1GYK3 10766696 Ki = 1.2 nM T76685 C8C6XK 10788693 Ki = 60.39 nM T76685 CI71YU 10789819 Ki = 1727 nM T76685 CV6A0K 10790480 Ki = 1119.4 nM T76685 C7WKY6 10807814 Ki = 434 nM T76685 C6XQA9 10812269 Ki > 10000 nM T76685 CN7T5O 10813167 Ki = 81.47 nM T76685 CRI9J2 10833730 Ki = 0.2 nM T76685 C8LF3D 10858553 Ki > 10000 nM T76685 C3TC7H 10871668 Ki > 10000 nM T76685 CK8MY5 10895601 Ki = 3700 nM T76685 CSG5H6 10902223 Ki > 10000 nM T76685 C1Q6BG 10906799 Ki = 162 nM T76685 C8SL5H 10928335 Ki = 24 nM T76685 CKT6I1 10950375 Ki = 1.8 nM T76685 CK6O4D 10972872 Ki = 56.9 nM T76685 CKX4U3 10982154 Ki = 374.1 nM T76685 C2XHD6 10982174 Ki = 0.4467 nM T76685 CJC9K4 11005810 IC50 = 6090 nM T76685 CCI2L6 11045217 Ki > 10000 nM T76685 C6LM0G 11048627 Ki = 7.8 nM T76685 C1S7MK 11048823 Ki = 32.3 nM T76685 CI8A6B 11076506 Ki > 10000 nM T76685 C9E2AP 11152300 Ki = 1600 nM T76685 CA79PI 11153626 Ki = 1 nM T76685 CF1DO0 11153651 EC50 = 6.31 nM T76685 CB47FY 11154357 EC50 > 3162.28 nM T76685 CA5OX2 11154964 Ki > 10000 nM T76685 CTN10X 11155520 Ki = 55 nM T76685 CMB65D 11157249 Ki = 589 nM T76685 CS92VB 11167681 IC50 = 26 nM T76685 CNI54S 11167736 IC50 = 0.47 nM T76685 CAP2S3 11168529 Ki = 23 nM T76685 C9S7TH 11169137 Ki = 724 nM T76685 C3HNI5 11178712 IC50 = 5.3 nM T76685 CW8V3S 11179949 Ki = 35.9 nM T76685 C8VWL5 11179964 Ki = 255 nM T76685 CTZ9G1 11180291 IC50 = 0.77 nM T76685 CJ9U8Q 11185771 Ki > 10000 nM T76685 C92AOP 11187538 Ki = 4780 nM T76685 CT8XE9 11188464 Ki = 48.6 nM T76685 CEST31 11188528 Ki = 79.7 nM T76685 CRK7V9 11189799 Ki = 828 nM T76685 C9E3HK 11190290 Ki = 1.5 nM T76685 C7VB3Y 11190694 Ki = 30 nM T76685 CM41GW 11192215 IC50 = 3.7 nM T76685 C59LVQ 11199737 EC50 > 3162.28 nM T76685 C9BOA6 11201612 EC50 = 10 nM T76685 CNF70Q 11201613 Ki = 1.585 nM T76685 CMXO58 11202164 Ki = 1 nM T76685 CB06ZT 11202865 IC50 = 1.3 nM T76685 C02GKP 11203203 Ki = 293 nM T76685 CY57AG 11212679 EC50 = 12.59 nM T76685 C73YFI 11213299 Ki = 106 nM T76685 CS2P5W 11213577 Ki = 214 nM T76685 C84YLO 11213961 IC50 = 0.73 nM T76685 C9BNR5 11224092 Ki = 2188 nM T76685 CEPJ47 11224779 Ki = 333 nM T76685 C7R2FT 11224783 Ki = 170 nM T76685 CLJH85 11226541 IC50 = 1.8 nM T76685 C7YUB3 11226720 Ki = 235 nM T76685 CQ4KW2 11235490 EC50 > 3162.28 nM T76685 C2AXJ6 11236772 Ki = 338 nM T76685 CQ36BE 11237017 Ki = 1412 nM T76685 CI8YG6 11237129 Ki = 13.9 nM T76685 CYE8Q0 11244542 Ki > 10000 nM T76685 C0UM9Z 11246347 Ki = 29.3 nM T76685 C8IQ7N 11247557 EC50 > 3162.28 nM T76685 C58AUX 11247638 Ki = 0.1 nM T76685 C7VTE6 11247889 Ki = 3.9 nM T76685 C5KOE4 11249677 Ki = 171 nM T76685 CRI87L 11259422 EC50 > 3162.28 nM T76685 CC4Q6B 11260007 IC50 = 120 nM T76685 CS9IP4 11260662 IC50 = 2.9 nM T76685 C2B6EC 11271934 Ki = 29 nM T76685 C9VEK5 11272442 Ki = 382 nM T76685 CEJ4I7 11283445 IC50 = 77 nM T76685 CWL54N 11293531 Ki = 94 nM T76685 CIA60C 11293559 Ki = 4 nM T76685 CC2J3W 11294205 Ki = 30 nM T76685 CI2HS8 11294476 IC50 = 1.3 nM T76685 C8E9AG 11294616 Ki = 36 nM T76685 CAB59V 11294643 Ki = 22.9 nM T76685 CZY4N1 11294721 Ki = 75.4 nM T76685 CL8FI9 11295086 Ki = 584 nM T76685 CBE45P 11295405 Ki = 356 nM T76685 C1T9CA 11305400 Ki = 52 nM T76685 C6J3MW 11306088 Ki = 35 nM T76685 C8FS1B 11306174 Ki = 24.2 nM T76685 C4H5FT 11318758 IC50 = 24 nM T76685 CZ47EO 11318799 IC50 = 2 nM T76685 CKUA15 11327582 EC50 > 3162.28 nM T76685 CBQO71 11328829 Ki = 3630 nM T76685 C9NW2C 11329073 Ki = 399 nM T76685 C8OAS0 11329521 IC50 = 1.8 nM T76685 CN6G7L 11329858 Ki = 221 nM T76685 CT8G0R 11338511 Ki = 250 nM T76685 CTQE86 11340501 Ki = 15 nM T76685 C4J9LE 11341568 IC50 = 46 nM T76685 C4G2KL 11349671 EC50 > 3162.28 nM T76685 C9UGA8 11349894 Ki = 2089 nM T76685 CDL7Q2 11352827 Ki = 993 nM T76685 C8AT6N 11363773 Ki = 894 nM T76685 COH57K 11373894 EC50 = 6.31 nM T76685 CQ26XK 11374417 Ki = 0.6 nM T76685 C0GP5M 11374894 Ki > 1000 nM T76685 C2SZV5 11375130 Ki = 27 nM T76685 CFA54H 11375615 Ki = 60 nM T76685 C7I9QK 11384486 Ki = 1.3 nM T76685 C8AZP3 11386027 Ki = 64 nM T76685 CB1T7I 11386417 Ki = 34 nM T76685 C7ZY4I 11386749 IC50 = 15 nM T76685 CJT18C 11387407 Ki = 1820 nM T76685 CB26AX 11391631 Ki > 10000 nM T76685 C4KX0N 11397179 Ki = 119 nM T76685 C37COB 11407971 Ki = 1 nM T76685 CD49YO 11408036 Ki = 1.7 nM T76685 CMSQ29 11408073 Ki = 3801 nM T76685 C4VPC8 11408345 Ki = 70.6 nM T76685 C2SWB7 11408408 Ki = 2193 nM T76685 CBN67Q 11408950 Ki = 14 nM T76685 CO6Z0Q 11409827 Ki = 36.5 nM T76685 CE7B0I 11410344 IC50 = 2.3 nM T76685 CY2ZI0 11413953 Ki = 6210 nM T76685 CJS85R 11429594 Ki = 45 nM T76685 CUSQ84 11430331 EC50 > 3162.28 nM T76685 C36OGJ 11432207 IC50 = 0.8 nM T76685 CFC95Y 11432710 IC50 = 0.9 nM T76685 C35TRL 11443469 IC50 = 24 nM T76685 CUN08B 11444148 IC50 = 32 nM T76685 CU2P3D 11451762 Ki = 34.9 nM T76685 C0MVE4 11452784 EC50 = 19.95 nM T76685 CE42DM 11453673 EC50 = 10 nM T76685 CQUG13 11454267 IC50 = 110 nM T76685 CAE92D 11454736 Ki = 54.2 nM T76685 CP3V7Z 11464072 Ki > 10000 nM T76685 C28OZA 11464704 Ki = 0.1 nM T76685 CV1M4Y 11466901 Ki = 1738 nM T76685 C4R5FJ 11467430 IC50 = 2.3 nM T76685 CFT60D 11475997 Ki = 3180 nM T76685 C61OKL 11476787 Ki = 403 nM T76685 CGC2Z6 11477574 IC50 = 96 nM T76685 CKP92B 11488130 Ki = 871 nM T76685 CO8H9L 11488131 Ki = 0.7 nM T76685 C9D2PH 11488705 IC50 = 0.7 nM T76685 C0CD5I 11489517 Ki = 6.28 nM T76685 C0VYA5 11493699 Ki = 1300 nM T76685 CQO3I6 11493987 Ki > 10000 nM T76685 CH0R5A 11494137 Ki = 245.47 nM T76685 CAR63Q 11494221 IC50 = 6.1 nM T76685 CN86KZ 11494391 Ki > 10000 nM T76685 CRLQ46 11494777 IC50 = 1400 nM T76685 CH79ND 11495004 Ki < 10000 nM T76685 C5B6XG 11495398 Ki = 210 nM T76685 C0C2AR 11495877 EC50 = 23 nM T76685 CJ1OG8 11496202 Ki = 59 nM T76685 CN3K8T 11496328 Ki = 75 nM T76685 CBD28Z 11496638 Ki = 24 nM T76685 CCQ85R 11501072 Ki = 38.9 nM T76685 CTYJ07 11501580 EC50 = 6300 nM T76685 C9Q0WB 11502034 Ki = 143 nM T76685 C1Z9YC 11502689 Ki = 1130 nM T76685 C0ZKG3 11504660 EC50 = 510 nM T76685 CNM0C3 11507880 Ki > 10000 nM T76685 CV8I4Q 11507883 Ki > 10000 nM T76685 CCDQ14 11508636 Ki = 91.2 nM T76685 C47RUL 11508949 Ki = 39.81 nM T76685 C1TC7Y 11510814 EC50 = 1000 nM T76685 CJ48YV 11515193 Ki > 10000 nM T76685 C1SF2Q 11515395 Ki = 676.08 nM T76685 C4U2YJ 11515910 Ki = 350 nM T76685 CDT27M 11516830 Ki > 10000 nM T76685 CB03ES 11517940 Ki > 10000 nM T76685 C23UNF 11517964 Ki = 77 nM T76685 C5DQ1X 11519312 Ki > 10000 nM T76685 CXI1O0 11522517 Ki = 660 nM T76685 CA5J2Z 11522912 Ki > 10000 nM T76685 C2YZM1 11522943 Ki = 380 nM T76685 CMEY72 11523234 Ki = 362 nM T76685 C20FDW 11524622 Ki > 10000 nM T76685 CAJO54 11525340 Ki = 5000 nM T76685 C3IGT1 11526889 Ki = 0.1995 nM T76685 CA7LK1 11529923 Ki = 630 nM T76685 CYR8X5 11530502 Ki = 204 nM T76685 C2Z3BK 11531885 Ki = 1900 nM T76685 CAN23D 11532254 EC50 = 1.4 nM T76685 CQ8L3J 11532557 Ki > 1000 nM T76685 C2UF3G 11533229 Ki = 5500 nM T76685 CK53RQ 11537652 Ki = 5.495 nM T76685 CVTA54 11537904 Ki = 790 nM T76685 C2C7YA 11541635 Ki = 2500 nM T76685 CSH2A1 11544639 EC50 = 4 nM T76685 CU49XP 11545113 Ki = 3360 nM T76685 CD1QL5 11546775 Ki = 1095 nM T76685 CC82RN 11548366 Ki > 10000 nM T76685 C6O3BK 11548933 Ki = 0.11 nM T76685 CB1DF3 11551160 Ki = 707.95 nM T76685 CTS15V 11551962 Ki = 2200 nM T76685 CNHP10 11552423 Ki > 3467.37 nM T76685 CQW9O7 11553971 Ki > 4040 nM T76685 CD3Q7W 11555661 Ki = 3000 nM T76685 C6GF0S 11559386 Ki = 14.79 nM T76685 CCB6F1 11559434 Ki = 27.54 nM T76685 CV06DX 11559474 Ki = 2951 nM T76685 CVX3N5 11559687 Ki = 2137.96 nM T76685 CT0YQ3 11560122 IC50 = 3600 nM T76685 C31FJV 11560244 Ki = 42 nM T76685 CON1Q8 11560246 Ki = 1925 nM T76685 CYUF67 11560249 EC50 = 3.84 nM T76685 CT5M4C 11560535 Ki > 10000 nM T76685 C5LVX9 11569155 Ki = 12500 nM T76685 C2N1IT 11569628 Ki = 3450 nM T76685 C3XD0O 11573397 Ki = 720 nM T76685 C5Y2NL 11574170 Ki > 10000 nM T76685 C0BT9C 11574627 Ki = 237 nM T76685 CS2T3B 11574895 IC50 = 10 nM T76685 COD9C6 11574958 Ki = 4250 nM T76685 CGF9C0 11575063 Ki = 800 nM T76685 C9JS7A 11576961 Ki = 280 nM T76685 C3VA1R 11580465 EC50 = 1881 nM T76685 CBS81K 11581197 Ki = 388 nM T76685 CCM0H1 11582155 Ki = 2000 nM T76685 CBF4O5 11583616 IC50 = 50.2 nM T76685 C3M6LW 11588379 Ki > 10000 nM T76685 C1H8NL 11589048 Ki = 1445.44 nM T76685 C0WK9H 11589652 EC50 = 10 nM T76685 C4WHZ5 11591162 EC50 = 133.9 nM T76685 C4EA7K 11595816 Ki = 44.67 nM T76685 CWV6T3 11595817 Ki = 1090 nM T76685 C0HFJ8 11597339 Ki > 1000 nM T76685 CF8L2I 11597475 Ki = 234 nM T76685 CU37FZ 11597700 Ki = 3000 nM T76685 C4CN3F 11601669 Ki = 14710 nM T76685 CU4I5W 11602703 Ki = 168 nM T76685 C0R1NH 11603123 Ki = 280 nM T76685 C4TN2S 11603482 IC50 = 31 nM T76685 CXL1Q2 11604689 EC50 = 37 nM T76685 CV43ZN 11605290 Ki > 10000 nM T76685 CJ18MB 11606800 Ki = 0.5012 nM T76685 C62OPJ 11609691 Ki = 309.03 nM T76685 C3FZJ9 11610001 Ki = 147.91 nM T76685 CMZ06K 11610023 Ki = 556 nM T76685 CN5U8O 11610189 EC50 = 79 nM T76685 CGZ98H 11611505 EC50 = 260 nM T76685 CRF2D3 11612574 Ki = 155 nM T76685 CV4K9F 11616911 Ki = 210 nM T76685 CW1M9F 11617449 IC50 = 220 nM T76685 CESR67 11617925 Ki = 9.3 nM T76685 CZ5FG6 11618026 Ki = 158 nM T76685 C8J9QA 11618679 Ki = 323 nM T76685 CH0I6J 11620691 IC50 = 40.7 nM T76685 C23WZM 11625937 Ki = 130 nM T76685 C14MPD 11626933 Ki = 3300 nM T76685 C8R1OK 11632670 Ki = 25 nM T76685 CA7K6Y 11638547 Ki > 10000 nM T76685 C6ZU0J 11640292 Ki = 105 nM T76685 C5K9JX 11641397 Ki = 16.1 nM T76685 CP1X4A 11646462 Ki = 13.8 nM T76685 C5BGP4 11648386 Ki = 39 nM T76685 C8Q0BW 11648843 Ki < 10000 nM T76685 C2IJK0 11653150 Ki = 180 nM T76685 CNOU53 11653233 Ki = 8.26 nM T76685 CYD30X 11653936 IC50 = 10 nM T76685 CS97YD 11654299 Ki = 460 nM T76685 C52VFG 11654304 Ki = 5.2 nM T76685 C1Q3HS 11655065 EC50 = 170 nM T76685 CWNX26 11659823 Ki = 80 nM T76685 C7ZI9D 11660288 Ki > 10000 nM T76685 CF59VR 11660635 Ki = 1995.26 nM T76685 C7N8JK 11660978 Ki = 4083 nM T76685 C7S9QI 11661782 Ki = 631 nM T76685 CF3D9J 11663483 EC50 = 1250 nM T76685 C7YDT1 11664479 Ki = 0.062 nM T76685 CD8EV7 11666821 Ki > 10000 nM T76685 CIX9F1 11667698 Ki > 10000 nM T76685 CYR0S8 11668868 Ki > 10000 nM T76685 CE7J1F 11669478 Ki = 33 nM T76685 CB7U5E 11670454 EC50 = 450 nM T76685 C59LNI 11673821 Ki = 2137.96 nM T76685 CP5SQ2 11675463 Ki = 1045 nM T76685 CM4OQ3 11675994 Ki = 11.7 nM T76685 C0NOQ3 11676975 Ki = 986 nM T76685 C1YVP6 11677439 EC50 = 540 nM T76685 C15MYH 11682550 Ki = 316 nM T76685 CO0Z4M 11683132 Ki = 1300 nM T76685 CYJ2U8 11683348 Ki > 10000 nM T76685 CEJ3R7 11683612 EC50 = 40 nM T76685 CCS3N5 11685395 Ki = 0.2512 nM T76685 CLB8K0 11688907 Ki = 691.83 nM T76685 CG8ZF9 11689178 Ki > 10000 nM T76685 C3WBU8 11689242 EC50 = 10000 nM T76685 CBW6K3 11689539 Ki = 1285 nM T76685 C1TI6L 11693193 Ki = 0.1259 nM T76685 C4CBE3 11695365 Ki > 10000 nM T76685 CSNO87 11696383 Ki < 10000 nM T76685 CMA60S 11696747 IC50 = 91 nM T76685 CZS68I 11697361 Ki = 1.7 nM T76685 C1ZUT0 11698933 Ki = 180 nM T76685 CI98GT 11699838 Ki = 0.1995 nM T76685 CXRS16 11703427 Ki = 11.7 nM T76685 C53ZLN 11705255 Ki = 152 nM T76685 CK7Z6O 11706218 IC50 = 35.8 nM T76685 CHN43G 11706783 Ki = 0.1259 nM T76685 CGI8A7 11708992 Ki > 10000 nM T76685 C2CX7N 11709987 Ki = 8430 nM T76685 CO40LS 11710271 Ki = 1154 nM T76685 CJE5D9 11712296 Ki = 141 nM T76685 CH7F8G 11713563 Ki = 2750 nM T76685 CQZ7T6 11716831 Ki = 213.8 nM T76685 CWRB76 11718456 Ki = 196 nM T76685 CY7KA2 11719546 Ki = 58 nM T76685 CE2H4Y 11719679 Ki = 1400 nM T76685 CV71DR 11725464 Ki = 2.9 nM T76685 C3L6FB 11748721 Ki >= 10000 nM T76685 CZ24IB 11752020 Ki = 1778 nM T76685 C09WKR 11755189 Ki = 0.1 nM T76685 C6AXN2 11756059 IC50 = 1.2 nM T76685 CAG2F1 11756523 Ki = 70.3 nM T76685 CGT70D 11758013 IC50 = 25 nM T76685 C7L0UM 11784543 Ki = 172 nM T76685 C8K4IE 11785274 IC50 = 35 nM T76685 C9K5HX 11785374 Ki = 21.8 nM T76685 C09CSH 11785582 Ki = 18 nM T76685 CP30IU 11785628 IC50 = 20 nM T76685 CE2DN3 11785870 Ki > 10000 nM T76685 C5MKE2 11794382 Ki = 13 nM T76685 CE9S1F 11800601 Ki = 19 nM T76685 CO7P6C 11842620 Ki = 43.8 nM T76685 CP2B0N 11851013 EC50 = 195 nM T76685 CQU9T1 11853103 Ki = 51 nM T76685 C3UQT0 11853349 Ki = 115 nM T76685 C8VK4D 11853588 Ki = 320 nM T76685 CFE9W6 11853590 Ki = 36 nM T76685 CUT8M5 11853591 Ki = 239 nM T76685 CBS7M9 11853844 EC50 = 11 nM T76685 C9IZT5 11854098 EC50 = 60 nM T76685 C3XF8V 11854101 EC50 = 5 nM T76685 CZ1G4T 11854358 EC50 = 115 nM T76685 COJ31I 11854359 Ki = 9 nM T76685 CLJ61F 11854361 Ki = 56 nM T76685 C4X2VS 11854364 EC50 = 5423 nM T76685 CDC1F6 11854609 EC50 > 14000 nM T76685 CCP14M 11854610 EC50 = 1360 nM T76685 C6OE1S 11856743 Ki = 15 nM T76685 C8TW9D 11856745 Ki = 58 nM T76685 CG70OF 11857227 Ki = 46 nM T76685 CPB2N7 11949613 Ki = 0.91 nM T76685 CL6Z1P 11949889 Ki = 51.1 nM T76685 CNW8M4 11950060 Ki = 10.6 nM T76685 C9EN7I 11950589 Ki = 51.6 nM T76685 CF7I2Q 11950590 Ki = 58.7 nM T76685 C89NBK 11950958 IC50 = 395 nM T76685 C0RNE1 11951124 EC50 = 3.9 nM T76685 CM0YF9 11951128 Ki = 67.7 nM T76685 CBV53O 11951300 Ki = 122 nM T76685 CGHC56 11951302 Ki = 5.1 nM T76685 C74VTU 11951655 Ki = 42.8 nM T76685 C1MTD0 11951656 Ki = 18.5 nM T76685 CFNY34 11951657 Ki = 23.6 nM T76685 C0DEG8 11951661 Ki = 40.2 nM T76685 CHVG30 11952383 Ki = 12.4 nM T76685 C4UOH8 11988884 Ki = 210 nM T76685 C1NKY7 11989761 Ki = 12 nM T76685 C4I9PA 11995515 Ki = 11 nM T76685 C43IFS 11995516 Ki = 4.7 nM T76685 C0FMG3 11996213 Ki = 4887 nM T76685 C68UFD 11996214 Ki > 10000 nM T76685 CY5VJ7 11996215 Ki > 1000 nM T76685 C3U2ZK 11996349 Ki > 10000 nM T76685 CDBZ94 11996350 Ki > 10000 nM T76685 CJO56E 11996351 Ki = 1422 nM T76685 CS34AL 11998407 Ki = 1.66 nM T76685 CZ6T5F 12000747 Ki = 57 nM T76685 C5KR9H 12000834 Ki = 0.75 nM T76685 CHC8O9 12000836 Ki = 0.04 nM T76685 C6RO3B 12000837 Ki = 0.11 nM T76685 CAQH93 12000925 Ki = 1 nM T76685 C9TMC1 12000926 Ki = 0.12 nM T76685 C53JEN 12000927 Ki = 0.25 nM T76685 CGN62B 12001013 Ki = 0.11 nM T76685 CLHV82 12146781 Ki > 5000 nM T76685 C5IL3V 12146783 Ki > 5000 nM T76685 C2U1FT 12147317 Ki = 5495 nM T76685 CRO26B 12471990 Ki > 10000 nM T76685 CEZD35 12971995 EC50 > 10000 nM T76685 CPD42A 13188551 Ki = 621 nM T76685 C9MQO2 14135316 IC50 = 1392 nM T76685 CF3W4S 14135317 IC50 = 184 nM T76685 C2TY8N 14135320 IC50 = 2400 nM T76685 CKP12X 14589394 Ki = 43 nM T76685 CF1EO5 14852550 Ki > 10000 nM T76685 C9C0DT 14898643 Ki > 10000 nM T76685 C5RCD3 14898644 Ki = 1340 nM T76685 C7Q8HG 14950683 Ki > 10000 nM T76685 CG49IS 14950684 Ki > 10000 nM T76685 CLK42M 14950685 Ki > 10000 nM T76685 CD13NW 14950686 Ki > 10000 nM T76685 C5THR8 15000083 Ki = 2.24 nM T76685 CP86TW 15000084 Ki = 628 nM T76685 CVGI15 15169782 IC50 = 0.32 nM T76685 C39MRN 15262805 Ki > 10000 nM T76685 CB0I3R 15341903 Ki = 3600 nM T76685 CIEM61 15481172 Ki = 243.8 nM T76685 CV25BT 15603837 Ki = 0.7 nM T76685 CGHE06 15953828 EC50 = 7943.28 nM T76685 C6NL8T 15991674 Ki = 77 nM T76685 CWP5Q0 15991676 Ki = 79 nM T76685 C20ZAI 15998061 Ki = 97 nM T76685 CX2CF4 15998383 Ki = 58 nM T76685 C0PU4I 15998702 Ki = 90 nM T76685 CP1X7K 16000037 EC50 = 500 nM T76685 CD6A0U 16004749 Ki = 0.1 nM T76685 CUSP63 16038085 IC50 = 2.4 nM T76685 CL9U8F 16045225 EC50 = 19.95 nM T76685 CC6O9T 16045226 Ki = 3.981 nM T76685 CJ78MO 16045297 Ki = 3.981 nM T76685 CM6FA4 16045299 EC50 = 50.12 nM T76685 C1AK4B 16049170 Ki = 0.1995 nM T76685 CZ7E3U 16067273 Ki > 10000 nM T76685 C1ST9R 16086925 Ki = 17 nM T76685 C4FY6M 16086929 Ki = 213 nM T76685 CJLP39 16086930 Ki = 30 nM T76685 C1R4QA 16098312 IC50 = 48 nM T76685 CCU10Q 16098313 IC50 = 13 nM T76685 C8JMW2 16098324 IC50 = 3 nM T76685 COK4S9 16098325 IC50 = 170 nM T76685 CJ27GS 16098334 IC50 = 1.5 nM T76685 CMET59 16098335 IC50 = 18 nM T76685 C0U3AZ 16098336 IC50 = 1.6 nM T76685 CM1PN6 16098337 IC50 = 1.8 nM T76685 C65WRB 16098343 IC50 = 1.3 nM T76685 CTHC39 16098344 IC50 = 0.54 nM T76685 CTZ95W 16098380 IC50 = 2 nM T76685 C4H5XE 16098381 IC50 = 1.1 nM T76685 C59CTW 16098382 IC50 = 19 nM T76685 CYN40W 16102907 Ki = 1.5 nM T76685 CIY74P 16223890 IC50 = 79.43 nM T76685 CGO03E 16224088 IC50 = 50.12 nM T76685 CDEL38 16224294 IC50 = 63.1 nM T76685 C7RO9Q 16226526 Ki = 1.259 nM T76685 CMH38I 16367681 Ki > 10000 nM T76685 C9APD3 16482860 EC50 > 10000 nM T76685 C3GN7A 16644329 Ki > 10000 nM T76685 CLY6K7 16659101 Ki = 2.2 nM T76685 C0WS7R 16659585 Ki = 0.37 nM T76685 CZ4H6L 16661349 Ki = 0.31 nM T76685 CAP57L 16661352 Ki = 0.01 nM T76685 C02TQV 16661501 Ki = 0.3162 nM T76685 CP98MW 16661502 Ki = 0.22 nM T76685 CK6RG8 16661654 Ki = 0.2512 nM T76685 C0L1OU 16661657 Ki = 0.1995 nM T76685 CZQ6R1 16661658 Ki = 0.3162 nM T76685 C6PBE3 16661819 Ki = 0.1 nM T76685 C8EK4I 16725534 EC50 = 320 nM T76685 C2F5LA 16737690 EC50 = 11 nM T76685 CHU72I 16738321 IC50 = 2.4 nM T76685 CY32BQ 16738395 IC50 > 6700 nM T76685 CGC6A8 16739312 IC50 = 2.8 nM T76685 CDN1E2 16748196 IC50 = 0.9 nM T76685 C5YF3B 16748318 IC50 = 0.9 nM T76685 CQP48T 16752691 IC50 = 4760 nM T76685 CK8M6J 16866369 EC50 = 17100 nM T76685 C28ZHR 17450266 Ki = 1900 nM T76685 C6JFW2 17592519 Ki > 10000 nM T76685 C9UGI2 17754357 Ki = 270 nM T76685 CEL3S7 17757539 Ki = 190 nM T76685 CVA94G 17955242 Ki = 240 nM T76685 C8WBK9 17984783 EC50 > 3162.28 nM T76685 CD9T6M 17984800 EC50 > 3162.28 nM T76685 CGV6D9 18106804 IC50 = 3162.28 nM T76685 CY7RP4 18407247 Ki = 52.6 nM T76685 C51JGA 18839400 Ki > 20000 nM T76685 CD89PR 19438815 Ki = 3363 nM T76685 C4H3AL 19868648 Ki = 2630 nM T76685 CJ2IL9 20386375 Ki > 3000 nM T76685 CATF15 21064882 Ki = 5.984 nM T76685 C7HIG9 21087760 Ki = 11 nM T76685 C0YC6G 21815908 Ki > 10000 nM T76685 CTL0C7 21858022 Ki > 10000 nM T76685 CF2S3C 21858023 Ki > 10000 nM T76685 C3YPZ2 21868807 Ki = 2.5 nM T76685 CBHZ92 21948978 Ki = 4.9 nM T76685 C7FC9A 21948995 Ki = 8.2 nM T76685 C8BW6H 21948996 Ki = 34 nM T76685 C94KPY 21949023 Ki = 14 nM T76685 C6N2GY 21949029 Ki = 12.2 nM T76685 C6F5VU 21949048 Ki = 66 nM T76685 C1OW2Z 21949050 Ki = 10 nM T76685 CJAZ80 21949054 Ki = 19 nM T76685 C45PAW 21984801 IC50 = 1.7 nM T76685 CZFS96 21984889 IC50 = 0.4 nM T76685 CT41MV 22038458 IC50 = 6.8 nM T76685 C8CO1J 22038459 Ki = 7.5 nM T76685 C6Y3AE 22038471 Ki = 74 nM T76685 C0JYB2 22038476 Ki > 2500 nM T76685 CP6E8S 22038485 IC50 = 67 nM T76685 C4NT8D 22038499 Ki = 10 nM T76685 CG3WD1 22038512 Ki = 4.1 nM T76685 CS50IQ 22038518 IC50 = 9.3 nM T76685 C6F5VP 22038520 IC50 = 17 nM T76685 CJ6HK9 22038546 Ki = 20 nM T76685 CMW59D 22181270 Ki > 5000 nM T76685 CFI69E 22181275 Ki > 5000 nM T76685 C0QOK7 22181282 Ki > 5000 nM T76685 CL52WO 22181288 Ki > 5000 nM T76685 C84HYE 22181294 Ki = 3475 nM T76685 CL45HJ 22181304 EC50 = 3235.94 nM T76685 C8OGN3 22181310 Ki > 5000 nM T76685 CSW3J7 22181316 Ki > 5000 nM T76685 CQRK86 22181322 Ki > 5000 nM T76685 CGC04B 22181344 Ki > 5000 nM T76685 C19BHA 22181345 Ki > 5000 nM T76685 C4S5NI 22181387 Ki > 5000 nM T76685 CX68DC 22181394 Ki > 4600 nM T76685 C9FX1Q 22181403 Ki > 5000 nM T76685 CX1U8F 22181408 Ki > 5000 nM T76685 CO87EI 22181435 Ki > 5000 nM T76685 CU61ZM 22266537 Ki > 5000 nM T76685 C7K3PT 22267343 Ki = 30 nM T76685 C6WLG2 22267384 Ki = 231 nM T76685 CUV02J 22267389 Ki = 60 nM T76685 CLI1M8 22267402 Ki = 223 nM T76685 C78LFV 22267403 Ki = 209 nM T76685 CIH20L 22285476 Ki = 22 nM T76685 CEI1J0 22285530 Ki = 1100 nM T76685 CSE31H 22285546 Ki = 130 nM T76685 C9O5TA 22422463 Ki = 198 nM T76685 C26KER 22422464 Ki = 58 nM T76685 C64NHO 22422466 Ki = 62 nM T76685 C1U4XQ 22431127 EC50 > 1000 nM T76685 C27SAH 22474540 EC50 = 420 nM T76685 CT8ZJ7 22475020 Ki = 4 nM T76685 CU83CN 22475030 Ki = 1 nM T76685 CT75AN 22475055 EC50 = 11 nM T76685 C6ZP8D 22475058 Ki = 30 nM T76685 C0N7IH 22475064 Ki = 216 nM T76685 CF9XZ1 22475102 Ki = 7 nM T76685 CH90RJ 22475113 EC50 = 2 nM T76685 CML7G3 22475120 Ki = 873 nM T76685 C09YAM 22475130 EC50 = 4 nM T76685 CTN92D 22475161 Ki = 277 nM T76685 CN9V2P 22475173 Ki = 18 nM T76685 C5ZM9W 22475232 Ki = 3 nM T76685 C40QAV 22475238 EC50 = 3 nM T76685 CX38ZN 22848569 Ki = 2600 nM T76685 CV2E0N 22969459 Ki = 1000 nM T76685 CK92XJ 23231044 Ki > 1000 nM T76685 C1ZT0J 23231127 Ki = 197 nM T76685 CNC4V7 23232560 Ki = 713 nM T76685 C0RL6E 23281241 Ki = 196 nM T76685 CJO3Z6 23328304 Ki = 16.6 nM T76685 C5OWG2 23398409 Ki = 18 nM T76685 C9H8QR 23398410 Ki = 6.3 nM T76685 CI0WV8 23398424 Ki = 6.9 nM T76685 CW1K2E 23398425 Ki = 97 nM T76685 CC5RT9 23398426 Ki = 75 nM T76685 C87MCO 23398428 Ki = 18 nM T76685 CHD4B5 23398430 Ki = 17 nM T76685 CU8I1Z 23398439 Ki = 2.2 nM T76685 CXDB37 23555594 Ki > 10000 nM T76685 CVB8K1 23555598 Ki = 336000 nM T76685 COB53R 23587763 Ki = 19 nM T76685 C2MC4Q 23588031 Ki = 322 nM T76685 C82JLB 23620581 Ki = 1906 nM T76685 CX8MY0 23626079 Ki = 1400 nM T76685 C8IVH5 23628267 Ki = 370 nM T76685 C3M9DF 23635640 Ki > 3000 nM T76685 CGN80J 23643046 Ki = 4400 nM T76685 CJ0QV7 23654188 Ki = 51 nM T76685 CMC87P 23654862 Ki = 3 nM T76685 C1LVE4 23656391 Ki = 1500 nM T76685 CA0VJ4 23730229 Ki = 150 nM T76685 CTKS21 23848377 Ki = 1800 nM T76685 CY48RZ 23968873 Ki = 2860 nM T76685 C52FSE 24096428 Ki = 0.77 nM T76685 CBU1K9 24125805 EC50 = 1174 nM T76685 C0DN4V 24180486 IC50 = 1700 nM T76685 CBXC05 24424330 IC50 = 0.58 nM T76685 C2CV7N 24467372 Ki = 450 nM T76685 CIP5B0 24748172 Ki = 27 nM T76685 C42DBF 24748217 Ki = 3008 nM T76685 CVNT09 24763642 IC50 = 4000 nM T76685 CT4SJ0 24766011 Ki > 10000 nM T76685 CFN89K 24768454 Ki > 2820 nM T76685 CNC6R4 24768455 Ki > 2820 nM T76685 CUE3X8 24768456 Ki > 2820 nM T76685 C5W8OH 24768457 Ki = 280 nM T76685 C7XE2U 24768458 Ki = 2820 nM T76685 CGF2B5 24768459 Ki = 280 nM T76685 CVD3X5 24768460 Ki = 110 nM T76685 CW35HD 24768461 Ki = 110 nM T76685 CC28YT 24768462 Ki = 2820 nM T76685 CU5P9T 24768463 Ki > 2820 nM T76685 CY3CP1 24768464 Ki = 2820 nM T76685 C8G6CH 24768465 Ki = 1850 nM T76685 CBU2P6 24768466 Ki = 37 nM T76685 C80IVA 24768467 Ki = 56 nM T76685 CFN6B5 24768468 Ki = 38 nM T76685 C5S0WL 24768469 Ki = 28 nM T76685 C61ELO 24768470 Ki = 42 nM T76685 CS6UN4 24768471 Ki = 28 nM T76685 CX79AV 24768472 Ki = 35 nM T76685 CSM3C5 24768473 Ki = 5.6 nM T76685 CR63JT 24768474 Ki = 28 nM T76685 C4CKN2 24768475 Ki = 280 nM T76685 CGZ9X6 24768476 Ki = 14 nM T76685 C8I4XR 24768477 Ki = 2800 nM T76685 C4K6QC 24768478 Ki > 2820 nM T76685 C09CZR 24768479 Ki = 2800 nM T76685 C1PR3H 24768480 Ki = 1600 nM T76685 C69VXF 24768481 Ki = 1600 nM T76685 CPBI12 24768482 Ki = 35 nM T76685 CWO6X4 24768483 Ki = 35 nM T76685 C6GKY8 24768484 Ki = 1800 nM T76685 C8IS0O 24768485 Ki = 280 nM T76685 CVIH02 24768486 Ki = 110 nM T76685 CV6HK2 24768487 Ki = 28 nM T76685 CC1B9L 24768488 Ki = 66 nM T76685 CHQ5E7 24768489 Ki = 1202.26 nM T76685 CS94WN 24768490 Ki = 501.19 nM T76685 CX86RC 24768491 Ki = 1905.46 nM T76685 CR1N5H 24768492 Ki = 13 nM T76685 CGJ93M 24768493 Ki = 69.18 nM T76685 C95JFQ 24768494 Ki = 1258.93 nM T76685 CBA0J3 24768495 Ki = 2804 nM T76685 CIC1H5 24768496 Ki = 776.25 nM T76685 CZAT71 24768497 Ki = 395 nM T76685 C3UIX7 24768498 Ki = 28 nM T76685 CVGO46 24768499 Ki > 1000 nM T76685 CX5N8F 24768500 Ki < 10000 nM T76685 C4E0SL 24768501 Ki > 3467.37 nM T76685 CX9CH8 24768502 Ki < 10000 nM T76685 C6AR0N 24768503 Ki > 2187.76 nM T76685 C4U9RH 24768504 Ki = 4073.8 nM T76685 C6X8BW 24768505 Ki = 3310 nM T76685 C8DJL5 24768506 Ki > 10000 nM T76685 CT6OR5 24768507 Ki > 10000 nM T76685 C1I4VG 24768508 Ki = 1698.24 nM T76685 CXAD71 24768509 Ki = 1862.09 nM T76685 CQLB52 24768510 Ki = 31 nM T76685 CRIJ68 24768511 Ki > 1000 nM T76685 CCV3R8 24768512 Ki = 228 nM T76685 C3H6RV 24775060 IC50 = 0.59 nM T76685 C6NQZ2 24779702 Ki = 150 nM T76685 CGLZ78 24779731 IC50 = 3500 nM T76685 C02APD 24794709 EC50 = 1280 nM T76685 CI3SF5 24797443 Ki = 16.7 nM T76685 C5U7ST 24798011 IC50 = 0.55 nM T76685 C52FXR 24801854 EC50 > 20000 nM T76685 CY93EF 24809843 Ki = 8.55 nM T76685 C2NQ6G 24825767 Ki = 48 nM T76685 CYQF93 24828287 EC50 = 2 nM T76685 CC6M0Z 24828288 Ki > 1000 nM T76685 CB9R7H 24828424 Ki = 509 nM T76685 CK8JY2 24828561 Ki = 13 nM T76685 CG9AZ6 24828562 Ki = 35 nM T76685 C52OSW 24828563 Ki = 3.3 nM T76685 CH9P2T 24849046 Ki = 20 nM T76685 CIC0B1 24856117 EC50 = 1920 nM T76685 C60CQO 24856504 Ki = 374 nM T76685 CH1AO3 24856554 Ki = 34.3 nM T76685 CZ7PQ6 24856591 Ki = 305 nM T76685 C7WDN2 24856637 Ki = 23.6 nM T76685 CM35KT 24856919 Ki = 139 nM T76685 CQ7Z3J 24857160 Ki = 3035 nM T76685 CLN2Y9 24857341 Ki = 1657 nM T76685 C67SFU 24857887 Ki = 1459 nM T76685 CI9ZX3 24857902 Ki = 0.83 nM T76685 C8XSM0 24857903 Ki = 0.24 nM T76685 CR2LS5 24862715 Ki = 32 nM T76685 CLG5O2 24863156 Ki = 68 nM T76685 C3P4FQ 24863231 Ki = 6.4 nM T76685 CECW68 24863252 Ki = 2.8 nM T76685 C3IA4J 24863253 Ki = 3.13 nM T76685 CXA79O 24863254 Ki = 2.53 nM T76685 CTJ1M4 24863255 Ki = 18.8 nM T76685 CB0NW8 24863396 Ki = 44.9 nM T76685 CP4Z2L 24863434 Ki = 491 nM T76685 C8UVA9 24863530 Ki = 51 nM T76685 CL2B6W 24863531 Ki = 15.3 nM T76685 CI2QU4 24863532 Ki = 7.4 nM T76685 C7Y2GK 24863613 Ki = 3.26 nM T76685 CMT60O 24863702 EC50 = 3.981 nM T76685 CBI19Y 24863730 Ki = 27 nM T76685 C4QXJ2 24863966 Ki = 19.3 nM T76685 CFV5K0 24864017 Ki = 1.08 nM T76685 CBP1Y5 24865177 Ki = 2800 nM T76685 CIY6F4 24865179 Ki = 320 nM T76685 C2D0YB 24873535 Ki = 560 nM T76685 CA6IE3 24880842 IC50 = 82.9 nM T76685 CXV19G 24881409 Ki = 17.9 nM T76685 CF5KN2 24881410 Ki = 148 nM T76685 C1HA5X 24881411 Ki = 5.83 nM T76685 CB4OX6 24881412 Ki = 152 nM T76685 CX2QD9 24881413 Ki = 116 nM T76685 CJZ52T 24881469 Ki = 14.7 nM T76685 CV3QZ2 24884489 Ki = 3800 nM T76685 C5OZ6A 24884501 Ki = 640 nM T76685 C4D8UX 24884502 Ki = 470 nM T76685 C25XLM 24890016 Ki = 4.365 nM T76685 CPEX19 24890017 IC50 = 1.995 nM T76685 CCJT43 24890180 IC50 = 0.7586 nM T76685 CZ50UW 24890182 Ki = 0.3981 nM T76685 C36SBO 24890183 Ki = 0.7943 nM T76685 CYJ94H 24890184 IC50 = 0.7762 nM T76685 CNQ6I4 24894028 EC50 = 49 nM T76685 C3C0KP 24894134 EC50 = 1430 nM T76685 CQY82F 24896430 Ki = 93.66 nM T76685 CJ8AB7 24901353 Ki = 66.3 nM T76685 CD7MS4 24944801 EC50 = 0.6 nM T76685 CK69LX 24944970 EC50 = 1.1 nM T76685 CPT7H9 24944972 EC50 = 0.5 nM T76685 CPL3Z0 24944973 EC50 = 6 nM T76685 C4X2MJ 24945064 EC50 = 5 nM T76685 CYDQ21 24945068 EC50 = 2.5 nM T76685 C0FE9Y 24945315 EC50 = 1.5 nM T76685 C5OX2A 24945317 EC50 = 2 nM T76685 CO1X2F 24945479 EC50 = 0.5 nM T76685 C63YSA 24945480 EC50 = 0.3 nM T76685 C82FVN 24945555 EC50 = 40 nM T76685 CRY7Z6 24945559 EC50 = 2.8 nM T76685 C0H6RV 24945635 EC50 = 0.5 nM T76685 CZ9S0C 24945636 EC50 = 0.5 nM T76685 CY58XE 24945637 EC50 = 2.2 nM T76685 CL91UP 24945796 EC50 = 4.6 nM T76685 CR94OQ 24945940 EC50 > 20000 nM T76685 CRD1G9 24946653 EC50 = 14700 nM T76685 C7MU9F 24947740 EC50 > 20000 nM T76685 C0UBF7 24947741 EC50 > 20000 nM T76685 C65EYT 24947742 EC50 > 20000 nM T76685 C85NPW 24952500 Ki = 4300 nM T76685 CHPT23 24953766 Ki = 1320 nM T76685 C5RN6C 24956045 Ki = 2500 nM T76685 CBW53M 24969357 IC50 = 0.63 nM T76685 C8QV4P 24983869 IC50 = 27.5 nM T76685 CPD69M 24984020 IC50 = 60.4 nM T76685 CH56TG 24984021 IC50 = 10.5 nM T76685 CPTK86 24984022 EC50 = 24.5 nM T76685 C3O5QS 24984023 EC50 = 293.6 nM T76685 CO42TL 24984332 IC50 = 1.4 nM T76685 CR5MP8 24984333 IC50 = 6.1 nM T76685 CZ9DE6 24984334 EC50 = 57.4 nM T76685 COQC35 24984485 EC50 = 348.8 nM T76685 CS1OQ5 24984486 IC50 = 1.2 nM T76685 C7DSG8 24984487 IC50 = 2.3 nM T76685 C3BIU6 24990210 EC50 > 10000 nM T76685 CZD3W7 24992427 IC50 = 1.7 nM T76685 C9YMN0 24994351 IC50 = 23 nM T76685 C2T0PY 24994664 IC50 = 8.2 nM T76685 CY74AK 24994665 IC50 = 4.9 nM T76685 C7VBJ3 24994981 IC50 = 1.3 nM T76685 C5PUR9 24994982 IC50 = 0.3 nM T76685 CZK8C0 24995602 IC50 = 15 nM T76685 CUMS01 24995912 IC50 = 120 nM T76685 C62VTZ 24996234 IC50 = 47 nM T76685 C2R6OP 24996235 IC50 = 15 nM T76685 CU7I2A 24996238 IC50 = 1.9 nM T76685 C34XJW 24996239 IC50 = 3.2 nM T76685 C13YJI 24996565 IC50 = 110 nM T76685 CO28GC 25006298 EC50 = 63.1 nM T76685 C6DVL4 25006674 Ki = 6.31 nM T76685 C2FA0Q 25006675 EC50 = 199.53 nM T76685 CETJ60 25006676 Ki = 19.95 nM T76685 C1IB2D 25024104 IC50 = 0.1 nM T76685 CH38VJ 25024106 IC50 = 1.9 nM T76685 CBPF20 25024108 IC50 = 1.3 nM T76685 CAB98T 25030040 Ki = 27 nM T76685 C9QM2T 25030041 Ki > 1000 nM T76685 CW7Q0H 25030042 Ki = 503 nM T76685 C40QGK 25033663 Ki = 2100 nM T76685 CW1D6E 25033664 Ki = 30.5 nM T76685 CE14PW 25033665 Ki = 160 nM T76685 CBW5O1 25033667 Ki = 6.1 nM T76685 C1A0QO 25033736 Ki > 10000 nM T76685 C3L4UA 25033812 EC50 > 10000 nM T76685 C91HVB 25033813 EC50 > 10000 nM T76685 CBN0A5 25033871 EC50 > 10000 nM T76685 CG18DC 25033872 EC50 > 10000 nM T76685 C6JAL1 25033874 EC50 > 10000 nM T76685 C7G3DB 25033875 EC50 > 10000 nM T76685 CJD73T 25033876 EC50 > 1000 nM T76685 CTQ29P 25033938 EC50 = 709 nM T76685 CJ6S9L 25033939 EC50 > 1000 nM T76685 C06YNQ 25033940 EC50 = 0.9 nM T76685 CZND73 25033941 EC50 > 1000 nM T76685 CGX95B 25033942 EC50 = 2000 nM T76685 C2N9UG 25033943 EC50 > 10000 nM T76685 C2J1HF 25034003 EC50 > 1000 nM T76685 CJ6G8M 25034004 EC50 > 1000 nM T76685 CS9J8K 25034005 EC50 > 1000 nM T76685 CBY1G8 25034006 EC50 > 1000 nM T76685 C6RY5L 25034007 EC50 > 1000 nM T76685 CJR0I9 25034070 EC50 = 472 nM T76685 CF7UY4 25034071 EC50 = 990 nM T76685 C2LB0M 25034073 EC50 > 10000 nM T76685 COCB26 25034074 EC50 > 10000 nM T76685 CH09EK 25034075 EC50 > 1000 nM T76685 CJF6E7 25034136 EC50 > 10000 nM T76685 CY5RI2 25034137 EC50 = 330 nM T76685 CKBP28 25034138 EC50 > 1000 nM T76685 COJC54 25034139 EC50 > 1000 nM T76685 C0UG1V 25034140 EC50 > 1000 nM T76685 CSF9M3 25034141 EC50 = 211 nM T76685 C7H3LM 25034205 EC50 > 1000 nM T76685 CPO3V5 25034206 EC50 > 1000 nM T76685 C3RZ9W 25034207 EC50 > 1000 nM T76685 CHC78S 25034208 EC50 = 670 nM T76685 CCQ81R 25034209 EC50 = 220 nM T76685 CZ0JY9 25034273 EC50 = 610 nM T76685 CL45CE 25034494 Ki > 10000 nM T76685 CX6RJ8 25034551 Ki = 1220 nM T76685 CTZ5D6 25034552 Ki = 2680 nM T76685 CI6RK0 25034553 Ki = 696 nM T76685 CN37RQ 25034554 Ki = 640 nM T76685 CY8C3F 25034555 Ki > 10000 nM T76685 C7S6GR 25034601 Ki = 139.8 nM T76685 CA0M1S 25034602 Ki = 14.3 nM T76685 CH5CJ1 25034603 Ki = 29.7 nM T76685 C9FY7P 25034605 Ki = 5.3 nM T76685 CI9KQ0 25034658 Ki = 28 nM T76685 CVM70G 25034659 Ki = 2630 nM T76685 CTOK52 25034660 Ki = 2520 nM T76685 C8E4BW 25034661 Ki = 739 nM T76685 CW07TE 25034662 Ki = 996 nM T76685 CC14IN 25052853 IC50 = 13.9 nM T76685 C1FU9T 25052854 IC50 = 1.2 nM T76685 C8GU5B 25052855 IC50 = 57.9 nM T76685 C3E8XA 25052856 IC50 = 20.6 nM T76685 CHIM64 25052920 EC50 = 35.5 nM T76685 CF6GE2 25052921 IC50 = 24.2 nM T76685 COL92Y 25052922 IC50 = 1.3 nM T76685 CGUL19 25052923 IC50 = 3 nM T76685 CF6AI2 25052924 IC50 = 2.1 nM T76685 C15YEA 25052990 IC50 = 21.7 nM T76685 CM19FU 25052991 EC50 = 442.4 nM T76685 CU28VO 25052992 EC50 = 20.4 nM T76685 C01ADI 25052993 IC50 = 12.7 nM T76685 CS8C7R 25052995 EC50 = 142.7 nM T76685 C8CSV3 25053066 EC50 = 18.7 nM T76685 CQ36FL 25053067 IC50 = 7.9 nM T76685 C2YSM3 25053068 IC50 = 4.9 nM T76685 C1KZ0L 25053142 EC50 = 23 nM T76685 CI8LQ6 25053143 EC50 = 51.4 nM T76685 CX6F8W 25053144 IC50 = 1.7 nM T76685 CXFL75 25053145 IC50 = 2.6 nM T76685 CZ79SF 25053146 EC50 = 28.9 nM T76685 C4WK5U 25053215 EC50 = 104.8 nM T76685 CSB7F9 25053216 IC50 = 82.4 nM T76685 C09NVD 25061041 IC50 = 130 nM T76685 C7R6MK 25070947 EC50 > 5000 nM T76685 CV4OA6 25094334 EC50 > 10000 nM T76685 C30WTM 25094337 EC50 > 10000 nM T76685 CY1FJ2 25094429 IC50 = 28 nM T76685 C6FZD5 25094431 IC50 = 3 nM T76685 C4UI7C 25094433 IC50 = 5.9 nM T76685 C40JMD 25094607 EC50 = 5623 nM T76685 CS2LZ4 25094611 EC50 > 10000 nM T76685 C9ZTU4 25094701 IC50 = 1.1 nM T76685 C5VIP4 25094884 EC50 > 10000 nM T76685 CTQB05 25095249 IC50 = 3.2 nM T76685 CALF53 25095275 IC50 = 4.1 nM T76685 CIK3S2 25095276 IC50 = 8.5 nM T76685 C7MXU4 25095277 IC50 = 9.5 nM T76685 CF2XN3 25095509 IC50 = 8 nM T76685 CH0W1V 25095533 IC50 = 1.9 nM T76685 CO76PH 25095792 IC50 = 2.2 nM T76685 C3IF6X 25095795 IC50 = 2.7 nM T76685 CBK9R7 25096563 IC50 = 82 nM T76685 C9LUX8 25096565 IC50 = 7.5 nM T76685 CRQ67O 25096567 IC50 = 1.1 nM T76685 CDC4X6 25097842 IC50 = 40 nM T76685 C1QX9B 25098113 IC50 = 16 nM T76685 C51OER 25098115 IC50 = 190 nM T76685 C2H6NK 25098369 IC50 = 10 nM T76685 CE75CG 25098370 IC50 = 34 nM T76685 C50QHA 25107503 Ki = 16.9 nM T76685 C6ZWJ3 25107504 Ki = 17.4 nM T76685 CMX36H 25107505 Ki = 0.5 nM T76685 CHV9I0 25107506 Ki = 0.3 nM T76685 C02LQB 25113749 IC50 = 62.8 nM T76685 CG64CV 25132791 EC50 > 10000 nM T76685 CS0Z2Y 25140206 Ki = 2300 nM T76685 CPB4N3 25140358 Ki = 3100 nM T76685 CDXE43 25140500 Ki = 8400 nM T76685 C3F4ZI 25140502 Ki = 1700 nM T76685 C6K7FP 25141397 Ki = 7800 nM T76685 CI69GZ 25143721 IC50 > 1000 nM T76685 CK15AS 25154780 Ki = 3.4 nM T76685 CYB6T7 25159779 Ki = 1548.82 nM T76685 C9MHD4 25159780 Ki > 10000 nM T76685 CK3BJ0 25159912 Ki > 10000 nM T76685 C8IZO3 25159915 Ki > 10000 nM T76685 CJRM20 25160046 Ki > 10000 nM T76685 C4V8RQ 25160840 IC50 = 549.54 nM T76685 CZ47PT 25168164 Ki = 54 nM T76685 CMYQ85 25168165 Ki = 42 nM T76685 C42VOK 25168166 Ki = 88 nM T76685 C6AHF5 25174166 EC50 = 6.2 nM T76685 CL9I5F 25178127 Ki = 1400 nM T76685 CK6Z9J 25181419 EC50 = 12589.25 nM T76685 CB0F5Z 25181480 EC50 > 2000 nM T76685 CWRL74 25181481 EC50 > 2000 nM T76685 CB8Y4M 25185393 Ki = 16000 nM T76685 C9XF6D 25185396 Ki = 850 nM T76685 C4O3KW 25186235 Ki = 2600 nM T76685 C9U6BE 25186236 Ki = 1000 nM T76685 C17XTC 25186238 Ki = 1100 nM T76685 C75ZTH 25186506 Ki = 210 nM T76685 C1XWS8 25186507 Ki = 1100 nM T76685 CB8Y1X 25186511 Ki = 1300 nM T76685 CRS71Z 25190875 Ki = 1.7 nM T76685 C4AE8F 25190876 Ki = 1.5 nM T76685 CIR2T7 25190877 Ki = 1.7 nM T76685 C4XIE6 25190878 Ki = 1.1 nM T76685 CMZ83A 25190879 Ki = 1.5 nM T76685 CG49HK 25190880 Ki = 1.6 nM T76685 CO9Z1E 25194977 EC50 = 87 nM T76685 CDZ2C4 25194999 IC50 = 19.3 nM T76685 CIE12A 25195000 EC50 = 22 nM T76685 CRW89Y 25195006 EC50 > 1000 nM T76685 CL41UB 25195469 EC50 = 10 nM T76685 C19CNW 25196320 Ki = 44.5 nM T76685 C0MQ7R 25196433 Ki = 177 nM T76685 CHS15A 25196434 Ki = 24.5 nM T76685 C3F5HA 25196664 Ki = 655 nM T76685 CF2O6Z 25196665 Ki = 2.8 nM T76685 C58AOY 25196773 Ki = 7.1 nM T76685 CM5V0Q 25197117 Ki = 1440 nM T76685 CF0O3T 25197227 Ki = 53.7 nM T76685 CR7AX1 25206705 Ki = 4.7 nM T76685 CTL8N0 25211883 Ki = 3400 nM T76685 CO2M3A 25221005 Ki = 2173 nM T76685 C4E2ZV 25222459 Ki = 6957 nM T76685 CC9J8H 25222461 Ki = 857 nM T76685 CZW14V 25222465 Ki = 2343 nM T76685 C2S5OU 25222569 Ki = 4710 nM T76685 C5LIC2 25222673 Ki = 817 nM T76685 CJT9H6 25222679 Ki = 3303 nM T76685 CSY93X 25222681 Ki = 2273 nM T76685 CKMF58 25223972 Ki = 2800 nM T76685 CAH40Z 25224932 Ki = 5700 nM T76685 C0IXY5 25230443 EC50 = 7.943 nM T76685 CF57PX 25230523 EC50 = 3.981 nM T76685 CX8QD0 25256778 Ki > 1000 nM T76685 C8C9FR 25266087 Ki = 13 nM T76685 CCG5U7 25266088 Ki = 14 nM T76685 C4O5EJ 25266089 Ki = 131 nM T76685 CD3CV0 25266090 Ki = 2 nM T76685 C48NMS 25266427 Ki = 32 nM T76685 CK4GE8 25266428 Ki = 33 nM T76685 C2JU5Q 25266429 Ki > 10000 nM T76685 CZOH53 25266430 Ki > 1000 nM T76685 CR9IE1 25266770 Ki = 10.3 nM T76685 CMK28L 25434865 Ki = 270 nM T76685 CI2TB6 26202942 Ki = 91 nM T76685 C0O3XE 26551661 EC50 > 10000 nM T76685 C5HP3T 26778303 EC50 = 1500 nM T76685 CC50YQ 42596959 Ki = 0.1995 nM T76685 C1NKQ6 42605511 IC50 = 100 nM T76685 CQ2SB1 42605622 IC50 = 8.5 nM T76685 CG7M1N 42605623 IC50 = 26 nM T76685 CY61ZS 42605958 IC50 = 25 nM T76685 CC7W2P 42607000 IC50 > 1000 nM T76685 C9TL5Q 42607230 IC50 = 32 nM T76685 CS4O0I 42607232 IC50 = 32 nM T76685 CK82HB 42617975 Ki = 61 nM T76685 CDM67X 42617976 Ki = 4.7 nM T76685 CF3HW5 42617977 Ki = 2.5 nM T76685 CQ2NR6 42617978 Ki = 4.7 nM T76685 CO8TK1 42617979 Ki = 24 nM T76685 CE6T1R 42617980 Ki = 11 nM T76685 CGSL84 42617982 Ki = 83 nM T76685 C9QF7X 42617987 Ki > 10000 nM T76685 CYB0L5 42617988 Ki > 10000 nM T76685 CCU97D 42617993 Ki = 2.512 nM T76685 CQD1I4 42617994 Ki = 0.3162 nM T76685 CW26DC 42617995 Ki = 0.7943 nM T76685 C9P6KA 42617996 Ki = 25.12 nM T76685 C9JMT1 42617997 Ki = 1.585 nM T76685 CGX62U 42617998 Ki = 39.81 nM T76685 CT2R8P 42625198 Ki = 2880 nM T76685 C14VEA 42625199 Ki = 310 nM T76685 CVN5E0 42625200 Ki = 10000 nM T76685 CN4ZG2 42625201 Ki = 1995.26 nM T76685 CEYI79 42625202 Ki = 5.012 nM T76685 CV60EY 42625203 Ki = 19.95 nM T76685 C9AK1Y 42625283 Ki = 10000 nM T76685 CZEB13 42625284 Ki = 100 nM T76685 CK3J1B 42625285 Ki = 5011.87 nM T76685 CWL7K2 42625370 EC50 = 180 nM T76685 CCE0P4 42625371 EC50 = 600 nM T76685 C64NGW 42625462 EC50 = 1500 nM T76685 CY4WS2 42625463 EC50 = 1 nM T76685 C64OXN 42625464 IC50 = 0.1 nM T76685 CJ4U7V 42625465 IC50 = 6 nM T76685 C6WX3B 42625466 IC50 = 8 nM T76685 CL48RK 42625547 IC50 = 2 nM T76685 CV3FM2 42625548 IC50 = 4 nM T76685 CZ96KC 42625549 IC50 = 5 nM T76685 C1U5IS 42625550 IC50 = 1.5 nM T76685 C6OKJ2 42625551 IC50 = 0.6 nM T76685 C1W2DX 42625635 IC50 = 50 nM T76685 C9GPZ5 42625636 IC50 = 0.3 nM T76685 C4C5QJ 42625708 IC50 = 10 nM T76685 C42OKY 42625711 EC50 > 10000 nM T76685 COT09H 42625787 EC50 = 7 nM T76685 C68FRN 42625790 EC50 = 1500 nM T76685 CJ71PG 42625791 EC50 = 1 nM T76685 CZ7AY8 42625862 EC50 = 1.3 nM T76685 CJ9WS6 42625863 IC50 = 0.5 nM T76685 CN5P0D 42625864 IC50 = 0.3 nM T76685 C4QWO7 42625865 IC50 = 8 nM T76685 C5XVB9 42625945 IC50 = 8 nM T76685 C6WYS0 42625946 IC50 = 0.7 nM T76685 CHQG38 42625947 IC50 = 7 nM T76685 CZ4V2A 42625948 IC50 = 0.3 nM T76685 C2VA7M 42625949 IC50 = 9 nM T76685 CQ1YN9 42626020 IC50 = 20 nM T76685 CIS6H0 42626021 IC50 = 100 nM T76685 CB18AO 42626022 IC50 = 400 nM T76685 C7K6PG 42626023 IC50 = 3 nM T76685 CJ8LY0 42626024 IC50 = 0.2 nM T76685 CMDL90 42626165 Ki = 2410 nM T76685 CHM37O 42626166 Ki = 50.12 nM T76685 CK27OJ 42626167 Ki = 794.33 nM T76685 CU7MV0 42626168 Ki = 251.19 nM T76685 C4D9KY 42626169 Ki = 199.53 nM T76685 CT1MQ0 42626170 Ki = 158.49 nM T76685 CL32WK 42626231 Ki = 2300 nM T76685 C23GWK 42626232 Ki = 1000 nM T76685 CG9X6Q 42626233 Ki = 2820 nM T76685 CH20LC 42626378 Ki = 10000 nM T76685 CW31TV 42626379 Ki = 3070 nM T76685 C6JYX3 43161871 Ki > 10000 nM T76685 C2D7FZ 44006806 Ki > 10000 nM T76685 CB0FC6 44157583 Ki = 560 nM T76685 CLP5D9 44157661 Ki = 5600 nM T76685 CZ67SH 44157662 Ki = 1000 nM T76685 CDT5M6 44157663 Ki = 6947 nM T76685 CRU08O 44157743 Ki = 18 nM T76685 CFV76H 44157744 Ki = 1519 nM T76685 C3DW6E 44157745 Ki = 200 nM T76685 C38DTW 44160263 Ki = 4.7 nM T76685 CVK7D9 44176908 Ki = 0.23 nM T76685 C8GY4U 44177029 Ki = 291 nM T76685 CH1XK6 44177030 IC50 = 403 nM T76685 CBCZ24 44177031 Ki = 5.8 nM T76685 C56QUX 44177146 Ki = 56 nM T76685 CES0V9 44177147 Ki = 111 nM T76685 CNE39O 44177148 Ki = 103 nM T76685 C34VDU 44177149 Ki = 1.6 nM T76685 C1NX0K 44177150 Ki = 0.2 nM T76685 CRE02Z 44177151 Ki = 2.6 nM T76685 CB2SO4 44177259 Ki = 1.2 nM T76685 C1V0SA 44177261 Ki = 1.1 nM T76685 C06NFO 44177371 Ki = 2.3 nM T76685 CI51QM 44177373 Ki = 0.15 nM T76685 C9B5WI 44177474 Ki = 60 nM T76685 C32AWN 44177475 Ki = 5.9 nM T76685 CBZL51 44177476 Ki = 1.8 nM T76685 CUS85Q 44177477 Ki = 2.2 nM T76685 C7A3CG 44177478 Ki = 8.1 nM T76685 CW3DR7 44177572 Ki = 1.2 nM T76685 C70RHS 44177573 Ki = 3 nM T76685 CXS2P1 44191632 IC50 = 107 nM T76685 CA7R6C 44191633 IC50 = 1110.8 nM T76685 CG3K4M 44191634 IC50 = 95.2 nM T76685 CLU36Q 44191688 EC50 = 9.8 nM T76685 CCHU94 44191689 IC50 = 16.3 nM T76685 CD50QV 44191690 EC50 = 81 nM T76685 C36RIL 44191691 IC50 = 42.5 nM T76685 C10TVJ 44191692 IC50 = 53.4 nM T76685 CO2FX0 44191743 IC50 = 12.3 nM T76685 CTS48Z 44191747 IC50 = 54.7 nM T76685 CZC56D 44191748 IC50 = 853.6 nM T76685 CU6RC5 44191749 IC50 = 248.9 nM T76685 CGY34V 44191806 EC50 = 12.3 nM T76685 C70DKR 44191807 IC50 = 197 nM T76685 C8PVX1 44191808 IC50 = 325.1 nM T76685 C4UXE0 44191809 IC50 = 47.4 nM T76685 C4DGZ9 44191810 IC50 = 211.8 nM T76685 CIK5H6 44191811 EC50 = 8.5 nM T76685 C5P2OJ 44191879 IC50 = 43.9 nM T76685 CY0F4D 44191880 EC50 = 20.2 nM T76685 CNR43E 44191881 IC50 = 14.6 nM T76685 CXT7B3 44191882 IC50 = 33.6 nM T76685 CR7PU3 44191883 IC50 = 33.8 nM T76685 CMAI32 44191949 EC50 = 5.1 nM T76685 C91ESC 44206133 EC50 = 2.1 nM T76685 CQH87P 44208932 Ki = 0.4 nM T76685 C3QC1N 44222441 Ki = 2400 nM T76685 C56IMC 44227470 IC50 = 2200 nM T76685 C9L7YS 44227471 IC50 = 940 nM T76685 CWA6J4 44247588 Ki = 9.2 nM T76685 CDR70U 44248166 Ki > 10000 nM T76685 CWC41U 44249869 EC50 = 7500 nM T76685 C6YU1J 44270301 Ki = 11 nM T76685 CHG1V2 44270339 Ki = 41 nM T76685 CI5XK7 44270344 Ki = 78 nM T76685 C5G8KN 44270345 Ki = 33 nM T76685 CKM95E 44270348 Ki = 101 nM T76685 C3AKR2 44270350 Ki = 94 nM T76685 CQX6Z1 44270362 Ki = 770 nM T76685 CLK8H3 44270364 Ki = 66 nM T76685 CWEC61 44270366 Ki = 14 nM T76685 CE14YI 44270369 Ki = 91 nM T76685 C0ZT6C 44270381 Ki = 32 nM T76685 C4CNP5 44270387 Ki = 29 nM T76685 CPDF42 44270403 Ki = 164 nM T76685 C7YD6L 44270429 Ki = 137 nM T76685 C8U7NS 44270430 Ki = 270 nM T76685 C6H0GU 44270432 Ki = 13 nM T76685 CD4S6V 44270441 Ki = 350 nM T76685 CCF24O 44282227 Ki = 3564.5 nM T76685 C5TGZ3 44282229 Ki = 605.3 nM T76685 CK8WE0 44282240 Ki = 203.2 nM T76685 CKSU69 44282639 Ki = 81.8 nM T76685 C94SQU 44300691 Ki > 20000 nM T76685 CL56ZV 44300702 Ki = 1.82 nM T76685 CRT85E 44300711 Ki = 350.3 nM T76685 CZB85J 44306648 Ki = 24 nM T76685 C76TNB 44307202 Ki = 245 nM T76685 CF8YK9 44307203 Ki = 8 nM T76685 C3JNX8 44307335 Ki = 21.88 nM T76685 CXT78N 44311448 Ki = 0.82 nM T76685 C32MHP 44312382 Ki = 1720 nM T76685 C74YBQ 44312424 Ki = 10253 nM T76685 C5T8JH 44312516 Ki = 4610 nM T76685 C89OGD 44312517 Ki = 3193 nM T76685 CP61BT 44312518 Ki = 6680 nM T76685 CP2V5L 44312529 Ki = 2183 nM T76685 CC68OA 44312599 Ki = 2553 nM T76685 C5FWB9 44312617 Ki = 5570 nM T76685 CI5NA2 44312651 Ki > 20000 nM T76685 CB72ZP 44312667 Ki = 16800 nM T76685 C0AL9Q 44312685 Ki = 2043 nM T76685 C0JK2Z 44313787 Ki = 650 nM T76685 CUA6G2 44316548 Ki = 5700 nM T76685 C3LA0K 44335317 Ki = 19 nM T76685 CM6T0I 44340976 Ki = 41 nM T76685 CX47WB 44344143 Ki = 0.57 nM T76685 C82CWR 44344222 Ki = 67.6 nM T76685 C8D7CT 44344236 Ki = 17.3 nM T76685 CDKT47 44345983 Ki = 0.7079 nM T76685 CKQ25P 44346066 Ki = 1.259 nM T76685 C9UCS2 44347216 Ki = 389 nM T76685 C0KC4U 44347229 Ki = 233 nM T76685 CO5AL2 44347231 Ki = 185 nM T76685 CZIT27 44350184 Ki = 0.77 nM T76685 C34MKG 44350470 Ki = 1297 nM T76685 CPU9G7 44358262 Ki = 0.36 nM T76685 CV3TI8 44373439 Ki = 220 nM T76685 C5AN8D 44373477 Ki = 12200 nM T76685 C40ERA 44373478 Ki = 1470 nM T76685 CC7UM4 44390004 IC50 = 500 nM T76685 CET9Q3 44390008 IC50 = 2200 nM T76685 CK9UO3 44390012 IC50 = 260 nM T76685 C2V9BA 44390024 IC50 = 80 nM T76685 CI5V2A 44390033 IC50 = 470 nM T76685 C73YIX 44390041 IC50 = 1000 nM T76685 CL2UH5 44390048 IC50 = 70 nM T76685 CXN3U4 44390055 IC50 = 200 nM T76685 CZVP65 44390375 EC50 = 28 nM T76685 C5KLM6 44390379 IC50 = 7.2 nM T76685 CS3DC0 44390402 IC50 = 66 nM T76685 C31PSD 44390412 IC50 = 18 nM T76685 CA4YS5 44390436 IC50 = 530 nM T76685 C0A5GI 44390447 IC50 = 6000 nM T76685 C2Q1LA 44390452 IC50 = 3.4 nM T76685 CZA0R4 44390459 IC50 = 3.1 nM T76685 CLW94E 44390460 IC50 = 18 nM T76685 C7GM2T 44390461 IC50 = 2000 nM T76685 CG7DF6 44390472 IC50 = 1.8 nM T76685 CBO6U4 44390485 IC50 = 8 nM T76685 CM2O6B 44390495 IC50 = 2.7 nM T76685 C6UC4N 44390702 Ki = 884 nM T76685 CENW29 44390703 IC50 = 18 nM T76685 C3NHV9 44390709 IC50 = 460 nM T76685 C9HKY5 44390712 EC50 = 50 nM T76685 C67BOD 44390716 IC50 = 41 nM T76685 C2B1WP 44390719 Ki = 1173 nM T76685 C3XN7P 44390728 IC50 = 7 nM T76685 CKC15H 44390729 Ki = 10625 nM T76685 C02LAG 44390734 IC50 = 22 nM T76685 CQ6I5W 44390735 IC50 = 1300 nM T76685 C7W3OJ 44390736 IC50 = 52 nM T76685 CQ0DN3 44390738 Ki = 2309 nM T76685 C53RBG 44390741 Ki = 100000 nM T76685 C04SIE 44390743 IC50 = 3.5 nM T76685 C6XG7M 44390744 IC50 = 58 nM T76685 C1FIA4 44390747 IC50 = 1.4 nM T76685 CKD9E1 44390751 Ki = 478 nM T76685 CN3WO0 44390753 IC50 = 400 nM T76685 CIQK65 44390754 Ki = 1758 nM T76685 CALH43 44390757 IC50 = 6 nM T76685 C52QMB 44390767 Ki = 1129 nM T76685 CBL63F 44390779 Ki = 855 nM T76685 C73BJO 44390783 Ki = 1172 nM T76685 CZ1H2T 44390792 Ki = 1923 nM T76685 CD1MC3 44390793 Ki = 117 nM T76685 C97KBA 44390799 Ki = 84 nM T76685 CHL9X5 44390813 Ki = 79 nM T76685 CF6L5S 44390825 Ki = 1779 nM T76685 C0MDC5 44390826 Ki = 72089 nM T76685 CAJG23 44390833 Ki = 1968 nM T76685 C1K6TJ 44390834 Ki = 3559 nM T76685 C5S6ET 44399915 Ki = 3467 nM T76685 CYJ7C4 44403115 Ki = 32 nM T76685 C4OT7Z 44403122 Ki = 117 nM T76685 C5WRH0 44403130 Ki = 125 nM T76685 C5VZU3 44403136 Ki = 141 nM T76685 C0MON3 44403143 Ki = 832 nM T76685 CVL3S8 44405953 Ki = 500 nM T76685 CPW2Z0 44405961 Ki = 200 nM T76685 C91IGO 44405962 Ki = 400 nM T76685 CMTI01 44405963 Ki = 600 nM T76685 C49YTQ 44405990 Ki = 300 nM T76685 C2PMS0 44406005 Ki > 10000 nM T76685 C1OFV8 44406006 Ki > 10000 nM T76685 CPJ3Y5 44406010 Ki > 10000 nM T76685 C1R7KG 44406065 Ki > 10000 nM T76685 C0R8HJ 44406069 Ki > 10000 nM T76685 CDH69R 44406086 Ki > 10000 nM T76685 CIJ4D9 44406096 Ki > 10000 nM T76685 CVK9O1 44406098 Ki > 10000 nM T76685 CJ8DT5 44406099 Ki = 500 nM T76685 C61TBI 44406108 Ki = 150 nM T76685 C8UJV2 44406124 Ki > 10000 nM T76685 CRYI42 44406130 Ki > 10000 nM T76685 CH76JQ 44406131 Ki > 10000 nM T76685 CP5OK0 44406141 Ki > 10000 nM T76685 CM4XA8 44406146 Ki = 500 nM T76685 C0Q2HD 44406147 Ki = 600 nM T76685 CEKQ30 44407258 IC50 = 5.2 nM T76685 CZW8H2 44407272 IC50 = 55 nM T76685 C8MA5H 44407369 Ki = 6 nM T76685 CF7ZB6 44407448 Ki = 38 nM T76685 CWD09L 44407449 Ki = 28 nM T76685 CA5G6X 44407528 Ki = 0.6 nM T76685 CUF1I7 44407557 Ki = 3 nM T76685 CY71IC 44407587 Ki = 21 nM T76685 CP1A5X 44407637 Ki = 4 nM T76685 C4QK2S 44407664 Ki = 12 nM T76685 CRH53I 44407665 Ki = 26 nM T76685 CA59QM 44407775 Ki = 1.8 nM T76685 CT34OK 44407776 Ki = 2 nM T76685 CO2S4P 44407798 Ki = 4 nM T76685 CY0N7C 44409165 Ki = 119 nM T76685 CSD7I2 44409348 Ki = 95.49 nM T76685 CZ7BA2 44409357 Ki = 27.9 nM T76685 CA1P5Z 44409404 Ki = 57.54 nM T76685 C5A3IS 44413438 Ki = 570 nM T76685 CA8L5B 44417321 Ki = 31.3 nM T76685 CAX6Z0 44421552 EC50 = 700 nM T76685 CC0HV3 44421553 Ki = 500 nM T76685 CXKZ94 44424074 Ki = 130 nM T76685 CG1W7H 44424075 Ki = 16 nM T76685 C3BV5M 44424076 Ki = 510 nM T76685 CYR36J 44424077 Ki = 560 nM T76685 CO14IM 44424078 Ki = 2100 nM T76685 CTIA24 44424079 Ki = 60 nM T76685 CI1NQ7 44424080 Ki = 750 nM T76685 C7G4KI 44424081 Ki = 260 nM T76685 CES0M4 44424082 Ki = 310 nM T76685 CGFH81 44424083 Ki = 750 nM T76685 CO29QR 44424084 Ki = 2100 nM T76685 CJ5A9X 44424085 Ki = 2820 nM T76685 CF3WD9 44424086 Ki = 170 nM T76685 CSGH07 44424087 Ki = 13 nM T76685 C05HAK 44424088 Ki = 56 nM T76685 C3GSH8 44424089 IC50 > 10000 nM T76685 CTDP28 44424090 IC50 > 10000 nM T76685 CFV9N7 44424091 IC50 > 10000 nM T76685 C3C5MS 44424092 IC50 > 10000 nM T76685 CFQ5V1 44424093 IC50 > 10000 nM T76685 CI27OV 44424094 Ki = 5.2 nM T76685 CIU4A6 44425199 Ki = 1.9 nM T76685 CP12WA 44425200 Ki = 25 nM T76685 C6KM1T 44425201 Ki = 7.2 nM T76685 CHP8W3 44425202 Ki = 36 nM T76685 C7HFJ8 44425203 Ki = 4.6 nM T76685 C4DGX2 44425204 Ki = 9 nM T76685 CS1YB3 44425205 Ki = 20 nM T76685 C1BI8C 44425206 Ki = 21 nM T76685 CGL6W2 44425207 Ki = 39 nM T76685 CPMY09 44425208 Ki = 95 nM T76685 C5ZHM4 44425209 Ki = 17 nM T76685 C3ZM0V 44425210 Ki = 34 nM T76685 CN9JM3 44425211 Ki = 270 nM T76685 CFO96B 44425212 Ki = 940 nM T76685 C9J5UB 44425213 Ki = 620 nM T76685 C14FAI 44425214 Ki = 920 nM T76685 CT5P7G 44425215 Ki = 22 nM T76685 CU6T4P 44425216 Ki = 41 nM T76685 C5JI1B 44425218 Ki = 10 nM T76685 CD2S1V 44425219 Ki = 19 nM T76685 CV2CW6 44425947 IC50 = 0.3 nM T76685 CUZ52I 44425948 IC50 > 2000 nM T76685 C7K3VZ 44425951 IC50 > 2000 nM T76685 CC9S6T 44425955 IC50 = 75.2 nM T76685 CE5DV6 44425957 IC50 = 1677 nM T76685 CH31IY 44425960 IC50 = 9.7 nM T76685 C50VBY 44425967 IC50 = 12.3 nM T76685 C1RI4V 44425970 IC50 = 13.9 nM T76685 C85WXL 44425974 IC50 = 21.7 nM T76685 C2S4TA 44425977 IC50 = 10.7 nM T76685 C8TW0V 44425983 IC50 = 7.1 nM T76685 C29RVL 44425996 IC50 = 7.4 nM T76685 C3D6XU 44425998 IC50 = 29.8 nM T76685 C8N7SY 44425999 IC50 = 11.4 nM T76685 COY28R 44426001 IC50 > 2000 nM T76685 C7KDN1 44426002 IC50 = 16 nM T76685 CN91SE 44426003 IC50 = 3.2 nM T76685 CTE8S2 44426005 IC50 = 5.1 nM T76685 C1N8SB 44426006 IC50 = 23 nM T76685 C7BQ6P 44426008 IC50 = 21.1 nM T76685 CK1Q6C 44426009 IC50 = 15 nM T76685 C95NOX 44426010 IC50 = 20.9 nM T76685 C8N7RU 44426011 IC50 = 16 nM T76685 CA4TQ0 44426012 IC50 = 53.5 nM T76685 C3YPC6 44426013 IC50 = 15.4 nM T76685 CQ7DY8 44426014 IC50 = 19.3 nM T76685 C5UE3X 44426015 IC50 = 41.8 nM T76685 C4BS5C 44426016 IC50 = 845 nM T76685 C5TJ3O 44426017 IC50 = 282.2 nM T76685 CAO8I2 44426020 IC50 = 37.2 nM T76685 C4UF8W 44426021 IC50 = 44.1 nM T76685 CM7S4D 44426022 IC50 = 38.3 nM T76685 CG9ZO2 44426300 Ki = 7.5 nM T76685 CS35IZ 44426301 Ki > 2500 nM T76685 CF9L3K 44426302 Ki > 2500 nM T76685 C8KAG7 44426303 IC50 = 16 nM T76685 C9VSG0 44426304 Ki = 6 nM T76685 CB50SY 44426305 Ki = 7.9 nM T76685 CWJ70K 44426306 Ki = 9.8 nM T76685 CAL59I 44426307 Ki = 920 nM T76685 CVXM58 44426308 Ki > 2500 nM T76685 CC32WE 44426309 Ki = 5.5 nM T76685 C36GVI 44426310 IC50 = 12 nM T76685 CQW3N7 44426311 Ki = 450 nM T76685 COIX34 44426312 IC50 = 37 nM T76685 CY5ZI3 44426313 IC50 = 19 nM T76685 C81IPU 44426314 IC50 = 20 nM T76685 C0MQR7 44426315 IC50 = 23 nM T76685 CA5Z1L 44426316 Ki = 390 nM T76685 C2FUP6 44426317 Ki = 2.8 nM T76685 CRV2P9 44426318 Ki = 200 nM T76685 C1VI9P 44426319 IC50 = 22 nM T76685 CY57HT 44426320 IC50 = 40 nM T76685 C04SIN 44426321 Ki = 3.5 nM T76685 CQ5L7T 44426373 Ki = 2000 nM T76685 CMTL10 44426375 Ki > 10000 nM T76685 CR9NI6 44426377 Ki > 10000 nM T76685 C5PV6B 44426379 Ki = 2600 nM T76685 C08URI 44426380 Ki > 10000 nM T76685 CJ04FU 44426381 Ki > 10000 nM T76685 CPU6S7 44426382 Ki > 10000 nM T76685 CHEC87 44426383 Ki > 10000 nM T76685 C67YNR 44426384 Ki > 10000 nM T76685 C32KAL 44427439 IC50 = 1100 nM T76685 C9Z3RU 44427440 IC50 = 300 nM T76685 C4AY0T 44427441 IC50 = 48 nM T76685 CUXF91 44427442 IC50 = 160 nM T76685 CWA8H9 44427443 IC50 = 930 nM T76685 CG4LS0 44427444 IC50 = 25 nM T76685 CPI40O 44431923 Ki = 13 nM T76685 C7GN9T 44431924 Ki = 1.8 nM T76685 CVB6N4 44431929 Ki = 160 nM T76685 C4ADH8 44431933 Ki = 120 nM T76685 CY0M2C 44431937 Ki = 24 nM T76685 CS7B0G 44431938 Ki > 1000 nM T76685 CX25NO 44431942 Ki > 1000 nM T76685 C82TOK 44431943 Ki = 2200 nM T76685 CVH58M 44431945 Ki = 1100 nM T76685 C96LUC 44431947 Ki = 39 nM T76685 C9ED7S 44431948 Ki > 1000 nM T76685 CK85UD 44431950 Ki = 840 nM T76685 C6OR5Y 44431952 Ki = 96 nM T76685 C8PR4Q 44431955 Ki = 1.7 nM T76685 C5PS7M 44431956 Ki = 4.6 nM T76685 CY25PR 44431957 Ki = 49 nM T76685 C3Z4DM 44431958 Ki = 600 nM T76685 C7NWB8 44431960 Ki = 34 nM T76685 CRV32B 44431963 Ki = 1400 nM T76685 CP2H7G 44431970 Ki = 27 nM T76685 C0Q6OE 44431973 Ki > 1000 nM T76685 C0BZM8 44431974 Ki > 1000 nM T76685 CGY89J 44431978 Ki = 320 nM T76685 C61GOU 44431987 Ki = 2.7 nM T76685 CX96RE 44431989 Ki = 370 nM T76685 CP7H0J 44431992 Ki > 1000 nM T76685 C87AWH 44431996 Ki = 360 nM T76685 CUY71Q 44432000 Ki = 1500 nM T76685 C6PO4R 44432001 Ki > 1000 nM T76685 CW3GF1 44432004 Ki = 3900 nM T76685 CJH15F 44432311 Ki > 5000 nM T76685 C8L1GT 44432313 Ki = 541 nM T76685 C5W3KH 44432314 Ki = 100 nM T76685 CMC1L8 44432316 Ki = 1260 nM T76685 CX84NA 44432317 Ki = 13 nM T76685 CPN2C1 44432318 Ki = 108 nM T76685 CUBO91 44432319 Ki = 671 nM T76685 CB64PA 44432320 Ki = 95 nM T76685 C9RLQ8 44432321 Ki = 514 nM T76685 CZ35SY 44432322 Ki = 1730 nM T76685 CW0A7J 44432323 Ki = 173 nM T76685 C26SPZ 44432324 Ki = 358 nM T76685 CP09WF 44432325 Ki = 418 nM T76685 C4EL9R 44432340 Ki = 711 nM T76685 CLR7C4 44432342 Ki = 114 nM T76685 C2FOQ4 44432345 Ki = 243 nM T76685 CW8OK2 44432347 Ki = 15 nM T76685 C3EP2D 44432349 Ki = 396 nM T76685 CO7M3T 44432351 Ki = 763 nM T76685 C10FBU 44432352 Ki = 44 nM T76685 C5CB6D 44432354 Ki = 246 nM T76685 CLQ5E1 44432356 Ki = 85 nM T76685 CP4B1S 44435054 Ki = 630.96 nM T76685 CE2U9J 44435055 Ki = 753.5 nM T76685 C0KUC3 44435059 Ki = 255 nM T76685 CGY1K2 44435062 Ki = 316.23 nM T76685 CT2Z7E 44435067 Ki = 134.9 nM T76685 COZ3W7 44435074 Ki = 1258.93 nM T76685 C6P7SG 44435076 Ki = 58.68 nM T76685 C9DBI0 44435083 Ki = 660.69 nM T76685 CPTZ16 44435085 Ki = 189 nM T76685 CT28WO 44437774 Ki = 194.85 nM T76685 C4T6JW 44437777 Ki = 86.33 nM T76685 CKS32L 44437778 Ki = 78.97 nM T76685 C5UZQ7 44437779 Ki = 8.87 nM T76685 C6RI2M 44437780 Ki = 2.74 nM T76685 CB34DJ 44437781 Ki = 5.51 nM T76685 CE8V6J 44437782 Ki = 131.33 nM T76685 C28YNG 44440473 Ki = 119 nM T76685 CMF83A 44440474 Ki = 129 nM T76685 CHC18G 44440477 Ki = 1251 nM T76685 CT0N3M 44440478 Ki = 1273 nM T76685 C28KUL 44440479 Ki = 2749 nM T76685 CERD71 44440480 Ki = 60.7 nM T76685 C6F2UJ 44440484 Ki = 3.7 nM T76685 CR1O0G 44440485 Ki > 10000 nM T76685 C8UB9Q 44440486 Ki = 3953 nM T76685 C7FND5 44440488 Ki = 7 nM T76685 CPT59U 44440489 Ki = 17 nM T76685 C6LWK7 44440494 Ki = 0.9 nM T76685 CDK0A6 44440509 Ki = 1099 nM T76685 C6OF1S 44440511 Ki = 21 nM T76685 CHAK08 44440521 Ki = 4.1 nM T76685 C7FPV3 44440528 Ki = 22 nM T76685 C52ATD 44440529 Ki = 14.4 nM T76685 CW0DE4 44440530 Ki = 115 nM T76685 CHE1A9 44440531 Ki = 140 nM T76685 C4KCQ2 44440532 Ki = 136 nM T76685 CYG41O 44440533 Ki = 58 nM T76685 C41OEA 44440534 Ki = 192 nM T76685 CF3ZC9 44440710 Ki = 110 nM T76685 CJE7X5 44440711 Ki = 59 nM T76685 C9A5DR 44440712 Ki = 178 nM T76685 CE6O7S 44440713 Ki = 18 nM T76685 C1N3YK 44440714 Ki = 5 nM T76685 C0CSL4 44440715 Ki = 25 nM T76685 C1L5YI 44440716 Ki = 203 nM T76685 C5UJ7Q 44440717 Ki = 33 nM T76685 C26AOF 44440721 Ki = 300 nM T76685 C06DPY 44440739 Ki = 167 nM T76685 C7XL1E 44440740 Ki = 50 nM T76685 C30KSN 44440741 Ki = 238 nM T76685 C7FBQ9 44440744 Ki = 14 nM T76685 CM30GA 44440991 IC50 = 0.91 nM T76685 CW1AG3 44440992 IC50 = 25 nM T76685 C1W7FC 44440993 IC50 = 50 nM T76685 CB9AL1 44440994 IC50 = 89 nM T76685 C75IOU 44440995 IC50 = 19 nM T76685 CCWQ18 44440996 IC50 = 20 nM T76685 CE3PF2 44440997 IC50 = 108 nM T76685 CMG6T0 44440998 IC50 = 37 nM T76685 CH6U8V 44440999 IC50 = 3.8 nM T76685 CJ4MX0 44441001 IC50 = 12 nM T76685 CSG2D8 44441002 IC50 = 5.9 nM T76685 C3RC0D 44441003 IC50 = 44 nM T76685 C1A7ZY 44441004 IC50 = 39 nM T76685 CJTA08 44441005 IC50 = 27 nM T76685 C4B7IT 44441006 IC50 = 38 nM T76685 CQN50B 44441007 IC50 = 165 nM T76685 C8I1UG 44441008 IC50 = 11 nM T76685 CMO79B 44441009 IC50 = 3.5 nM T76685 CABT03 44441010 IC50 = 5.6 nM T76685 C7VL0N 44441011 IC50 = 80 nM T76685 C2RU3Y 44443139 IC50 = 53 nM T76685 CNBC42 44443143 IC50 = 1100 nM T76685 C7U1DE 44443144 IC50 = 140 nM T76685 C6P3MF 44443150 IC50 = 4100 nM T76685 CZU3M6 44443151 IC50 = 690 nM T76685 C0BMK4 44443156 IC50 = 19 nM T76685 C9LE0K 44443158 IC50 = 830 nM T76685 CY14CG 44443159 IC50 = 1500 nM T76685 CCK4Z5 44443160 IC50 = 1200 nM T76685 CHVC86 44443161 IC50 = 1900 nM T76685 CVY34E 44443162 IC50 > 10000 nM T76685 CH5J7Y 44443368 Ki = 20.1 nM T76685 C8P2BQ 44443370 Ki = 259 nM T76685 CY69LT 44443371 Ki > 8000 nM T76685 C7RJ8Z 44443372 Ki = 1811 nM T76685 CJ2KY6 44443373 Ki = 695 nM T76685 CKB28C 44443375 Ki = 658 nM T76685 C3X6WY 44443379 Ki = 279 nM T76685 C0Y5IS 44443394 Ki = 137 nM T76685 CE5YJ9 44443395 Ki = 195 nM T76685 C4T6WD 44443396 Ki = 2331 nM T76685 CB4X3O 44443398 Ki = 818 nM T76685 C8U6EH 44443400 Ki = 2914 nM T76685 CF4J1Q 44443401 Ki > 8000 nM T76685 CUHZ49 44443404 Ki = 2131 nM T76685 CSF47I 44443409 Ki = 7222 nM T76685 C68LRJ 44443410 Ki = 779 nM T76685 CY2EA4 44443414 Ki = 1473 nM T76685 C6FX1J 44443415 Ki = 973 nM T76685 C70JDW 44443417 Ki = 3021 nM T76685 CZEH01 44443422 Ki = 6183 nM T76685 C9AB0R 44443423 Ki = 263 nM T76685 CZ3NL8 44443425 Ki = 418 nM T76685 C9V7IM 44443426 Ki = 604 nM T76685 C1CJ9Y 44443427 Ki = 341 nM T76685 CK76YZ 44443428 Ki = 176 nM T76685 CAW0S5 44443429 Ki = 339 nM T76685 C3N7TI 44443430 Ki = 2742 nM T76685 CFMQ75 44443432 Ki = 1273 nM T76685 CF41HI 44444731 Ki > 5600 nM T76685 CDO2Y1 44444732 Ki = 170 nM T76685 C1N2HC 44444733 Ki = 2920 nM T76685 CM13FT 44444734 Ki = 17 nM T76685 CO40HV 44444735 Ki = 290 nM T76685 C95JLA 44444737 Ki = 5600 nM T76685 CUWH37 44444738 Ki = 620 nM T76685 C9H4MD 44444739 Ki = 560 nM T76685 CSE7K2 44444740 Ki > 5600 nM T76685 C28XNW 44444741 Ki = 2800 nM T76685 C8Z4VB 44444945 Ki = 14 nM T76685 CC6R1O 44444946 Ki = 10.9 nM T76685 C6ZFB9 44444947 Ki = 3.9 nM T76685 CWJ25A 44444948 Ki = 2.7 nM T76685 CA5P0S 44444949 Ki = 141 nM T76685 C7IX3A 44444950 Ki = 297 nM T76685 CRY47W 44448494 Ki > 10000 nM T76685 CA49WS 44448505 Ki > 10000 nM T76685 C6AY8U 44448506 Ki > 10000 nM T76685 C7ZJ9O 44448536 Ki > 10000 nM T76685 C72IYN 44448539 Ki > 10000 nM T76685 CZTQ62 44448540 Ki > 10000 nM T76685 C4G9YD 44448542 Ki > 10000 nM T76685 CBA36L 44448576 Ki > 10000 nM T76685 CSB9M8 44448577 Ki > 10000 nM T76685 C0J4VA 44448578 Ki > 10000 nM T76685 CGL3J5 44448579 Ki > 10000 nM T76685 COWF13 44448613 Ki > 10000 nM T76685 C7VGI3 44448615 Ki > 10000 nM T76685 CIR53D 44448618 Ki > 10000 nM T76685 CVB6E5 44448647 Ki > 10000 nM T76685 CS9YA3 44448648 Ki > 10000 nM T76685 C7JYR2 44448650 Ki > 10000 nM T76685 C4FXJ0 44449070 Ki = 1300 nM T76685 CRG1Z7 44449071 Ki > 1000 nM T76685 CCI20B 44449072 Ki = 540 nM T76685 C5T0BS 44449073 Ki = 470 nM T76685 CLG5M9 44449097 Ki = 310 nM T76685 CYN7U8 44449099 Ki = 50 nM T76685 C84CJE 44449124 Ki = 130 nM T76685 CQ4X9R 44449155 Ki = 93 nM T76685 C3X6IU 44449157 Ki = 110 nM T76685 CM4O5I 44449158 Ki > 1000 nM T76685 C75QPO 44449159 Ki = 89 nM T76685 C4YA1F 44449217 Ki = 1300 nM T76685 C4U1IW 44449219 Ki > 1000 nM T76685 CYQ15R 44449322 EC50 = 320 nM T76685 C3G5QB 44450408 Ki = 52.8 nM T76685 C5V3QC 44450418 Ki = 301.4 nM T76685 C50DPE 44450419 Ki = 451.5 nM T76685 C5NHR2 44450433 Ki = 46 nM T76685 C2OX1G 44450447 Ki = 839 nM T76685 CXGD98 44450450 Ki = 110 nM T76685 C8OHS5 44450451 Ki = 1500 nM T76685 CH10PO 44452652 IC50 = 870 nM T76685 CBJG30 44452653 IC50 = 760 nM T76685 C76GPX 44452677 IC50 = 810 nM T76685 C75KBE 44453101 IC50 = 3700 nM T76685 CCKA13 44453126 IC50 = 1300 nM T76685 C2R4WU 44454162 Ki = 172 nM T76685 C3CX0V 44475155 EC50 = 61.4 nM T76685 C8VJ5L 44475188 EC50 > 30000 nM T76685 CO42MQ 44475189 EC50 > 30000 nM T76685 CB93OS 44475190 EC50 > 10000 nM T76685 CKL9D6 44475191 EC50 = 25100 nM T76685 CZ4E7R 44475345 EC50 = 15800 nM T76685 CX8MZ5 44475348 EC50 = 10000 nM T76685 CZMG41 44475514 EC50 > 30000 nM T76685 CLF27M 44475515 EC50 > 30000 nM T76685 C8TKO9 44475665 EC50 > 30000 nM T76685 C4YJ7O 44475667 EC50 > 30000 nM T76685 CX9Y5J 44475668 EC50 = 4000 nM T76685 CNXU56 44475669 EC50 > 30000 nM T76685 C45KSU 44475670 EC50 = 6300 nM T76685 C37BCT 44476482 Ki = 2 nM T76685 CJXC18 44476564 Ki = 38.8 nM T76685 CMNK07 44476566 Ki = 7.6 nM T76685 CF6WL7 44476567 Ki = 55 nM T76685 COT18G 44482558 Ki < 10 nM T76685 CO3GJ9 44517703 Ki = 50 nM T76685 C1YJ6M 44517704 Ki = 3.4 nM T76685 CGK87Q 44555025 Ki = 4.7 nM T76685 C4RB7W 44555352 Ki = 7.6 nM T76685 CF8G9Y 44559754 IC50 = 41 nM T76685 CV0RU3 44560201 IC50 = 424 nM T76685 CJKY16 44560203 IC50 = 316 nM T76685 CL8M3P 44560218 IC50 = 128 nM T76685 CI0T8G 44560219 IC50 = 226 nM T76685 C2FCI9 44560231 IC50 = 441 nM T76685 CFP0N9 44560232 IC50 = 729 nM T76685 C4D9CJ 44560233 IC50 = 1040 nM T76685 CF2XA9 44560240 IC50 = 273 nM T76685 CB8T0A 44560241 IC50 = 443 nM T76685 C7O8DG 44560242 IC50 = 195 nM T76685 CD05GO 44560243 IC50 = 163 nM T76685 CL3DV8 44560269 IC50 = 340 nM T76685 C9W8VR 44560270 IC50 = 334 nM T76685 C0M2DU 44560271 IC50 = 186 nM T76685 CT98QB 44560272 IC50 = 204 nM T76685 C8UBN6 44561004 Ki > 5000 nM T76685 CU4SG5 44561005 Ki = 1209 nM T76685 CB25AC 44561006 Ki > 5000 nM T76685 CMDC01 44561007 Ki > 5000 nM T76685 C71HSJ 44561015 Ki = 13.7 nM T76685 CPTB84 44561045 Ki > 5000 nM T76685 COD91U 44561114 Ki > 5000 nM T76685 CMD3W0 44561115 Ki > 5000 nM T76685 CY36FG 44561116 Ki > 5000 nM T76685 C1W9IC 44561150 Ki > 5000 nM T76685 C08RTQ 44561151 Ki > 5000 nM T76685 CYFN50 44561189 Ki = 4679 nM T76685 CK3IH5 44561190 Ki > 5000 nM T76685 C9P8KC 44561230 Ki > 5000 nM T76685 CVD07Y 44561231 Ki > 5000 nM T76685 CKZS21 44561232 Ki = 4190 nM T76685 C4N9BV 44561233 Ki = 2396 nM T76685 C0O2ER 44561273 Ki > 5000 nM T76685 C13COW 44561274 Ki > 5000 nM T76685 CPG0S6 44561275 Ki = 2608 nM T76685 CB5S1Y 44561307 Ki > 5000 nM T76685 CG42HW 44561308 Ki > 5000 nM T76685 CD5O4Z 44561342 Ki > 5000 nM T76685 C0EC3G 44561343 Ki > 5000 nM T76685 CQDJ15 44561375 Ki = 2483 nM T76685 CI18KY 44561376 Ki > 5000 nM T76685 C3N6MT 44561377 Ki > 5000 nM T76685 CFL6K1 44561532 Ki = 3115 nM T76685 C1NKS2 44561533 Ki = 110 nM T76685 C80YSF 44561534 Ki = 406 nM T76685 CM1S2X 44561571 Ki = 4766 nM T76685 CUH92O 44561572 Ki > 5000 nM T76685 C9WP1L 44567376 IC50 = 798 nM T76685 C85QKG 44567397 IC50 = 49.4 nM T76685 CJIT49 44567398 IC50 = 146 nM T76685 C3WDR4 44567399 IC50 = 286 nM T76685 CIPL70 44569452 EC50 > 10000 nM T76685 C42IGT 44569453 EC50 = 82 nM T76685 C3S9KJ 44569454 EC50 = 1570 nM T76685 C1AL6B 44569455 EC50 > 10000 nM T76685 CDWS53 44569456 EC50 > 10000 nM T76685 C6Y0LF 44569505 EC50 > 2000 nM T76685 C9VLE7 44569506 EC50 > 1000 nM T76685 C3TO8N 44569507 EC50 > 1000 nM T76685 C7CRO4 44569508 EC50 > 1000 nM T76685 C91HRZ 44569553 EC50 > 10000 nM T76685 CTJR64 44569554 EC50 > 10000 nM T76685 C62ROA 44569555 EC50 > 10000 nM T76685 CX72NB 44569556 EC50 > 10000 nM T76685 CWT7A1 44569557 EC50 > 10000 nM T76685 C9MTC0 44569587 EC50 = 96 nM T76685 CRTA75 44569588 EC50 = 322 nM T76685 CUYD25 44569589 EC50 > 10000 nM T76685 CD6W1Y 44569590 EC50 > 10000 nM T76685 C92FOT 44569622 EC50 > 10000 nM T76685 CWQ1K2 44569623 EC50 = 1650 nM T76685 CUJ4A1 44569924 EC50 > 3162.28 nM T76685 C08SCG 44569925 EC50 > 3162.28 nM T76685 CJT9Q2 44569926 EC50 > 3162.28 nM T76685 CB5S9R 44569927 EC50 > 3162.28 nM T76685 C1HWD3 44570015 EC50 > 3162.28 nM T76685 CQ7XA5 44570119 EC50 > 3162.28 nM T76685 C5WLK8 44570120 EC50 > 3162.28 nM T76685 C1CO2M 44570121 EC50 > 3162.28 nM T76685 C34ZJI 44570122 EC50 > 3162.28 nM T76685 C1WN9J 44570165 EC50 > 3162.28 nM T76685 CM1I9W 44570166 EC50 > 3162.28 nM T76685 CCR56A 44570167 EC50 > 3162.28 nM T76685 CSE9N3 44570253 EC50 > 3162.28 nM T76685 CX9T2R 44570254 EC50 > 3162.28 nM T76685 CYOA27 44570255 EC50 > 3162.28 nM T76685 CP32DL 44570256 EC50 > 3162.28 nM T76685 CB4VL6 44570296 EC50 > 3162.28 nM T76685 C27RYN 44570535 EC50 > 3162.28 nM T76685 C40ZIV 44570573 EC50 > 3162.28 nM T76685 CDI76Z 44570574 EC50 > 3162.28 nM T76685 C3MY6V 44570575 EC50 > 3162.28 nM T76685 CT93YR 44570576 EC50 > 3162.28 nM T76685 CHR90O 44570577 EC50 > 3162.28 nM T76685 CVZ47U 44570611 EC50 > 3162.28 nM T76685 CS2G7D 44570612 EC50 > 3162.28 nM T76685 C5MIN6 44570613 EC50 > 3162.28 nM T76685 CXJN76 44571487 EC50 = 122 nM T76685 C5FR4V 44571527 EC50 = 216.3 nM T76685 C8NDA0 44571528 IC50 = 144.4 nM T76685 CGA62W 44571564 EC50 = 256.1 nM T76685 CNBW05 44571566 EC50 = 235.2 nM T76685 CBV09K 44571567 IC50 = 25.7 nM T76685 CYLG38 44571593 Ki = 49 nM T76685 C68APE 44571594 Ki = 31 nM T76685 C13FQU 44571595 Ki = 624 nM T76685 CJQC45 44571596 Ki = 515 nM T76685 CKB8D4 44571640 EC50 = 56.2 nM T76685 CX16CU 44571641 EC50 = 12.2 nM T76685 C7TC0V 44571642 EC50 = 17.8 nM T76685 CBS48G 44571676 Ki = 59 nM T76685 C7XF1J 44571677 Ki = 152 nM T76685 CKD2R0 44571678 Ki = 1 nM T76685 CCQR65 44571679 Ki = 0.9 nM T76685 CR10QM 44571680 Ki = 1 nM T76685 C32TAP 44571692 EC50 = 136.2 nM T76685 C8XGL2 44571725 Ki = 17 nM T76685 C0C9FB 44571726 Ki = 4.9 nM T76685 C4JAB8 44571727 Ki = 9.2 nM T76685 CN2T8Z 44571728 Ki = 14 nM T76685 C6HM3V 44571773 Ki = 4.9 nM T76685 CJ4AM7 44571774 Ki = 14 nM T76685 C8VM7B 44571775 Ki = 76 nM T76685 CC7I1B 44571776 Ki = 101 nM T76685 C2Q9CJ 44572101 IC50 = 4496.8 nM T76685 CT2K8N 44573966 IC50 = 398.11 nM T76685 CJMV73 44573967 IC50 = 776.25 nM T76685 CIWU28 44573968 IC50 = 2187.76 nM T76685 CDHA03 44574009 IC50 = 3467.37 nM T76685 CS42HA 44574010 IC50 = 6606.93 nM T76685 C24BJY 44574096 IC50 = 20.89 nM T76685 C6LTX4 44574097 IC50 = 1698.24 nM T76685 CQ67PU 44574098 IC50 = 2041.74 nM T76685 CPS52D 44574122 IC50 = 6.166 nM T76685 CQL80H 44574576 EC50 = 690 nM T76685 C2LG7H 44574577 EC50 = 800 nM T76685 CCVH32 44574623 EC50 = 1330 nM T76685 CQ76AC 44574665 IC50 = 1500 nM T76685 CM83FT 44574781 IC50 = 150 nM T76685 C9TZM7 44574993 IC50 = 100 nM T76685 CW8RY0 44576567 Ki = 2100 nM T76685 C3BA8P 44576568 IC50 > 10000 nM T76685 CJGC60 44576569 IC50 > 10000 nM T76685 COC9J6 44576570 IC50 > 10000 nM T76685 CVI5W4 44576588 IC50 > 10000 nM T76685 CJ8A9D 44576623 Ki = 2720 nM T76685 CQ7L2J 44576639 IC50 > 10000 nM T76685 CR14SW 44576640 Ki = 1480 nM T76685 CFW4H3 44576641 IC50 > 10000 nM T76685 C93RWF 44576654 Ki = 69 nM T76685 C0LP2G 44576658 Ki = 1.75 nM T76685 CX70KJ 44576659 Ki = 14.96 nM T76685 C4D8NU 44576660 Ki = 2.84 nM T76685 C8EQ0F 44576673 Ki = 3010 nM T76685 CQLC63 44576674 IC50 > 10000 nM T76685 CX6N2C 44576675 IC50 > 10000 nM T76685 CQV82A 44576683 Ki = 32.33 nM T76685 C3Q6PU 44576684 Ki = 9.81 nM T76685 CB7M6F 44576685 Ki = 0.67 nM T76685 CORN72 44576686 Ki = 0.87 nM T76685 CY94LQ 44576715 Ki = 1.2 nM T76685 C8THE4 44576716 Ki = 1.97 nM T76685 CNC54I 44576717 Ki = 0.8 nM T76685 CEG98D 44576969 Ki = 1730 nM T76685 C0SLX2 44577003 Ki = 1510 nM T76685 CY0S8V 44577004 IC50 > 10000 nM T76685 C1H6LE 44577006 IC50 > 10000 nM T76685 CFE0J9 44577551 EC50 = 15 nM T76685 C9GW1T 44577552 EC50 = 419 nM T76685 C6SC5G 44577607 EC50 = 96 nM T76685 C48TNK 44577700 EC50 = 2620 nM T76685 C3K5WB 44577701 EC50 = 951 nM T76685 CG4A6T 44577703 EC50 = 600 nM T76685 CIC7Q0 44578053 EC50 = 403 nM T76685 CBO9H2 44578091 EC50 = 1560 nM T76685 C6G5AM 44578092 EC50 = 1300 nM T76685 CC04VP 44578093 EC50 = 2230 nM T76685 CX3Y1N 44578140 EC50 > 2000 nM T76685 C1ART0 44578141 EC50 = 1270 nM T76685 C0HJZ8 44578142 EC50 = 1690 nM T76685 CA5R4C 44578214 EC50 = 910 nM T76685 CKA97I 44578215 EC50 = 722 nM T76685 CD79OE 44578574 Ki = 280 nM T76685 C7LRN5 44578575 Ki = 560 nM T76685 CD43MU 44578576 Ki = 2200 nM T76685 CBPI67 44578618 Ki = 560 nM T76685 CFXZ16 44578619 Ki = 220 nM T76685 C5MY0R 44578620 Ki = 560 nM T76685 C8C5XG 44578653 Ki = 560 nM T76685 C5NFK4 44578654 Ki = 560 nM T76685 CYF2L0 44578655 Ki = 560 nM T76685 CSX6U1 44578656 Ki = 900 nM T76685 C6DO8E 44578695 Ki = 2200 nM T76685 C8UP7T 44581023 Ki = 381 nM T76685 C7CNY2 44581106 Ki > 10000 nM T76685 C0UA7D 44581107 Ki = 5055 nM T76685 C21CLI 44582191 Ki = 24 nM T76685 CT0N5V 44582835 Ki = 3400 nM T76685 C7CK6B 44582862 EC50 > 10000 nM T76685 C5DC6O 44582872 EC50 > 10000 nM T76685 CA2CH8 44582883 EC50 = 8 nM T76685 CEJ81A 44582896 EC50 = 900 nM T76685 CVT0K8 44586998 EC50 = 850 nM T76685 CJ38WB 44586999 EC50 = 470 nM T76685 C9AKC5 44587055 EC50 = 810 nM T76685 C65SDP 44587305 Ki = 15 nM T76685 CP6T2X 44588588 Ki = 1900 nM T76685 CHI7K5 44588701 Ki = 6000 nM T76685 C21ZJU 44588702 Ki = 8600 nM T76685 CR1IM7 44591240 Ki = 510 nM T76685 C5P9YH 44591241 Ki = 750 nM T76685 C6N1BV 44591252 Ki = 540 nM T76685 CGH2M3 44591253 Ki = 790 nM T76685 CH3QA7 44591254 Ki = 1800 nM T76685 C1IS0P 44591270 Ki = 390 nM T76685 C6CK0Q 44591271 Ki = 200 nM T76685 C5TY6G 44591272 Ki = 260 nM T76685 C5OAG4 44591273 Ki = 130 nM T76685 CTN05S 44591293 Ki = 560 nM T76685 CX3J9M 44591294 Ki > 5000 nM T76685 CI4F5K 44591295 Ki = 140 nM T76685 CU2Z1B 44591296 Ki = 310 nM T76685 CB87ZC 44591297 Ki = 530 nM T76685 CZC2V8 44591328 Ki = 1100 nM T76685 C0RG5Z 44591329 Ki = 1100 nM T76685 C8EZ2F 44591330 Ki = 770 nM T76685 CFJ6T4 44591331 Ki = 270 nM T76685 C9VER2 44591332 Ki = 740 nM T76685 CB92EJ 44591350 Ki = 1400 nM T76685 C2VMW7 44591351 Ki = 6990 nM T76685 C5MY2H 44591352 Ki = 1200 nM T76685 CIZR27 44591353 Ki = 1200 nM T76685 C1GB8U 44591372 Ki = 1200 nM T76685 COL9S4 44591395 Ki = 2900 nM T76685 C3LF9C 44591610 IC50 = 316.23 nM T76685 CS3CO8 44591625 IC50 = 10 nM T76685 C3D6NC 44591626 IC50 = 2.512 nM T76685 CI1H3S 44591631 Ki = 30 nM T76685 CPD59V 44591648 IC50 = 6.31 nM T76685 C6NMS8 44591716 IC50 = 19.95 nM T76685 C0NJE8 44592106 Ki = 13.7 nM T76685 CQ45LI 44593416 Ki = 9.25 nM T76685 CU5QM9 44593417 Ki = 2.72 nM T76685 CUS0P8 44593426 Ki = 34.4 nM T76685 C96SDI 44593427 Ki = 11 nM T76685 CALE39 44593428 Ki = 1.85 nM T76685 COX3D7 44593429 Ki = 1.77 nM T76685 C3LH5A 44593430 Ki = 76.1 nM T76685 C6URQ2 44593432 Ki = 5.03 nM T76685 C6AKT4 44593433 Ki = 1.59 nM T76685 CC0ZX7 44593612 IC50 > 10000 nM T76685 CS16LT 44608360 Ki = 14.5 nM T76685 CH3K4A 44608519 Ki = 7.5 nM T76685 CU26YR 44608681 Ki = 42 nM T76685 CW9TR0 44608682 Ki = 140 nM T76685 CMC89D 44626286 Ki = 43 nM T76685 CL25CW 44626287 Ki = 74 nM T76685 CMS21C 44626293 Ki = 47 nM T76685 CW62LE 44626508 Ki > 10000 nM T76685 CHCX20 44626509 Ki > 10000 nM T76685 CWH62A 44626510 Ki > 10000 nM T76685 CF98KL 44626511 Ki > 10000 nM T76685 C4HA1P 44626512 Ki = 280 nM T76685 CP5D3I 44626513 Ki = 4265.8 nM T76685 CHQ34G 44626514 Ki = 91 nM T76685 CYB13E 44626619 Ki = 144.54 nM T76685 CLI40Y 44626620 Ki > 10000 nM T76685 C57FZK 44626621 Ki = 1819.7 nM T76685 CJLY69 44626623 Ki > 10000 nM T76685 C9VP2H 44626624 Ki = 2030 nM T76685 CM5Q6F 44626625 Ki = 47.86 nM T76685 C56HJF 44626626 Ki = 1900 nM T76685 CQ9ZE1 44626729 Ki > 10000 nM T76685 CQ90WV 44626834 Ki > 10000 nM T76685 CY4UX7 44627979 Ki > 10000 nM T76685 CN01CV 44627980 Ki = 1621.81 nM T76685 CONU92 44627981 Ki = 616 nM T76685 CVCP89 44627983 Ki > 10000 nM T76685 CH1S3P 44627984 Ki = 3057 nM T76685 CL2PS3 44628086 Ki = 131 nM T76685 C4VB5F 44628087 Ki = 61.66 nM T76685 CP2Y8T 44628090 Ki > 10000 nM T76685 CAL60M 44629129 Ki = 12.2 nM T76685 CN91XU 44806719 Ki > 10000 nM T76685 CD0B8E 45101490 EC50 = 0.9 nM T76685 C2TYD1 45254043 Ki = 500 nM T76685 C7QW2B 45256133 EC50 > 50000 nM T76685 CYU95D 45256135 EC50 > 20000 nM T76685 CBPO23 45267412 Ki = 1049 nM T76685 CDLT14 45268251 Ki = 1473 nM T76685 CIDM75 45269488 EC50 = 14000 nM T76685 C4CXU8 45272121 Ki = 1.3 nM T76685 CJK2T4 45272898 EC50 = 18000 nM T76685 CAMX32 45277748 Ki = 3.1 nM T76685 C6UVZ0 45277749 Ki = 5.9 nM T76685 CK5G2I 45277750 Ki = 2.5 nM T76685 CMO74A 45375898 EC50 = 10000 nM T76685 C2P7DZ 45482145 Ki = 20 nM T76685 CI2L3H 45482146 Ki = 70 nM T76685 C2RHP4 45482154 Ki = 120 nM T76685 C5AYP0 45482155 Ki = 96 nM T76685 CLY7J6 45482156 Ki = 90 nM T76685 CVX13E 45482170 Ki = 140 nM T76685 CLD6B9 45482181 Ki = 227 nM T76685 CN2D1B 45482194 Ki = 70 nM T76685 CP3A2G 45482195 Ki = 144 nM T76685 CS8IL1 45482196 Ki = 30 nM T76685 CRZ7E0 45482212 Ki = 157 nM T76685 C83GHF 45482213 Ki = 117 nM T76685 CPB4V3 45482221 Ki = 368 nM T76685 CKZD49 45482222 Ki = 112 nM T76685 C5V0BJ 45482230 Ki = 156 nM T76685 CDI5R8 45482231 Ki = 150 nM T76685 CC1N8T 45482236 Ki = 218 nM T76685 C71YGP 45482237 Ki = 84 nM T76685 CD8O6R 45482242 Ki = 56 nM T76685 C3FZ2G 45482253 Ki = 1300 nM T76685 CJS5B4 45482262 Ki > 2820 nM T76685 C4BMX6 45482263 Ki = 100 nM T76685 C0KX7R 45482264 Ki = 310 nM T76685 C69UKE 45482265 Ki = 948 nM T76685 C0SW4I 45482271 Ki = 390 nM T76685 C3WO9A 45482272 Ki = 380 nM T76685 C01KMJ 45482275 Ki = 36 nM T76685 CMZI72 45482276 Ki = 12 nM T76685 CY2C1A 45482277 Ki = 2100 nM T76685 CU2A6Y 45482278 Ki = 340 nM T76685 C97TZR 45482285 Ki = 240 nM T76685 C0RK2J 45482286 Ki = 50 nM T76685 CMLT59 45482287 Ki = 165 nM T76685 C8YK5V 45482288 Ki = 54 nM T76685 CM1QD0 45482290 Ki = 5.6 nM T76685 CB9F2E 45482291 Ki = 31 nM T76685 C9QCD0 45482292 Ki = 14 nM T76685 CLM52Q 45482293 Ki = 2400 nM T76685 CG8ME6 45482294 Ki = 5.6 nM T76685 CE0C1R 45482295 Ki = 99 nM T76685 C1IUF2 45482296 Ki = 41 nM T76685 C9NPK7 45482298 Ki = 560 nM T76685 CGDH61 45482299 Ki = 840 nM T76685 C8CNJ6 45482300 Ki = 56 nM T76685 C3CJY6 45482302 Ki = 80 nM T76685 CX1W2E 45482305 Ki = 345 nM T76685 CV2H0Q 45482306 Ki = 560 nM T76685 C7WH3G 45482308 Ki > 2820 nM T76685 CF5AU0 45482309 Ki = 56 nM T76685 CT61ZB 45482312 Ki = 80 nM T76685 CI4KQ8 45484652 Ki = 540 nM T76685 C80ZSJ 45484668 Ki = 1100 nM T76685 CWO0Z4 45484669 Ki = 110 nM T76685 C0US3O 45484688 Ki = 1400 nM T76685 C93GPE 45484689 Ki = 2100 nM T76685 CG5KM4 45484698 Ki = 9000 nM T76685 CR8OU6 45484699 Ki = 1700 nM T76685 CQ9E8H 45484714 Ki = 3900 nM T76685 C1TH8B 45484715 Ki > 5000 nM T76685 C4ENV9 45484721 Ki = 1300 nM T76685 CS4Z1M 45484728 Ki = 6300 nM T76685 C9IS4Y 45484737 Ki = 1600 nM T76685 C0L4KU 45484747 Ki = 130 nM T76685 CG8Q2A 45484758 Ki = 9 nM T76685 C8WN5C 45484794 Ki = 4.7 nM T76685 C4M2GB 45484803 Ki = 5 nM T76685 CXC8O9 45484808 Ki = 9 nM T76685 C6RZ1I 45484813 Ki = 7.9 nM T76685 CH53YJ 45484814 Ki = 3.8 nM T76685 C0VYP1 45486166 EC50 = 10000 nM T76685 C8RXB2 45486199 EC50 > 31622.78 nM T76685 CNKE85 45486200 EC50 > 31622.78 nM T76685 CIE6R2 45486207 EC50 > 31622.78 nM T76685 C7TQB2 45486215 EC50 = 10000 nM T76685 CT7D5W 45486221 EC50 > 31622.78 nM T76685 C9PR0W 45486227 EC50 > 31622.78 nM T76685 C0R2LC 45486228 Ki > 10000 nM T76685 C5XH8U 45486229 Ki = 4200 nM T76685 CF7DI2 45486232 Ki = 72.44 nM T76685 C5MGW3 45486233 Ki = 537.03 nM T76685 C28VPU 45486235 Ki > 10000 nM T76685 CMS0L5 45486237 Ki > 10000 nM T76685 C93XDH 45486386 Ki = 43 nM T76685 CX42VA 45486394 Ki = 31 nM T76685 CNDU21 45486467 Ki = 3.1 nM T76685 CG9D2X 45486479 Ki = 19 nM T76685 CBL5Q4 45486480 Ki = 9.6 nM T76685 CER4H7 45486486 Ki = 701 nM T76685 CNE83F 45486585 IC50 = 46.1 nM T76685 CL7O8R 45486588 IC50 = 17.9 nM T76685 CL2M1O 45486624 EC50 = 3.2 nM T76685 CZI3A7 45486625 IC50 = 12.2 nM T76685 CDZ06Y 45486626 IC50 = 37.7 nM T76685 C5LM1E 45486627 IC50 = 49 nM T76685 CFU06M 45486645 IC50 = 49.2 nM T76685 CX03TG 45487312 EC50 = 1.9 nM T76685 CO02JA 45487319 IC50 = 47.7 nM T76685 CR31BT 45487337 IC50 = 19.5 nM T76685 C4RWJ7 45487338 IC50 = 2982 nM T76685 C1HX4V 45487344 EC50 = 3.5 nM T76685 CDME83 45487345 IC50 = 132 nM T76685 CQ48YZ 45487350 IC50 = 136 nM T76685 C6MSZ4 45487367 IC50 = 186 nM T76685 C6QZT8 45487368 IC50 = 301 nM T76685 CYID78 45487377 IC50 = 203 nM T76685 CV8Y7U 45487389 IC50 = 97 nM T76685 CC5WX3 45487684 Ki = 1100 nM T76685 CJC8B3 45487735 EC50 > 30000 nM T76685 CA7H4J 45487736 EC50 > 30000 nM T76685 C5BD3E 45487753 EC50 > 30000 nM T76685 CXA9P3 45487780 Ki = 1800 nM T76685 C82GUQ 45504069 Ki = 288 nM T76685 CN31HO 46191641 EC50 > 31622.78 nM T76685 CME02J 46209990 IC50 = 2565 nM T76685 CS81HE 46216704 Ki = 3.8 nM T76685 C4SD8K 46216705 Ki = 9.1 nM T76685 C8TFL3 46216706 Ki = 6.3 nM T76685 C2VP6F 46216778 Ki = 5 nM T76685 CW4E2J 46220521 EC50 > 100000 nM T76685 CYQ03E 46224624 Ki = 1400 nM T76685 C3R0TH 46224630 Ki = 1800 nM T76685 CDS69K 46224634 Ki = 3400 nM T76685 C1UNT4 46224640 Ki = 3800 nM T76685 CS5TO6 46224659 Ki = 2100 nM T76685 C7X2AF 46224661 Ki = 1700 nM T76685 CBOD08 46224662 Ki = 650 nM T76685 C9E6XS 46224717 IC50 = 1.2 nM T76685 C5DR4L 46224718 IC50 = 5.8 nM T76685 C7OK0Q 46224719 IC50 = 2.6 nM T76685 CWR12J 46224720 IC50 = 4.1 nM T76685 CTQ2F3 46224773 IC50 = 4.2 nM T76685 CW7PG8 46224774 IC50 = 1.6 nM T76685 CP2Z3T 46224775 IC50 = 7 nM T76685 C87GHR 46224776 IC50 = 0.51 nM T76685 CC5J6U 46224814 IC50 = 0.7 nM T76685 CCX52N 46224815 IC50 = 5.6 nM T76685 C38IKB 46224921 IC50 = 11 nM T76685 C3TB8O 46224922 IC50 = 57 nM T76685 C27CZA 46224923 IC50 = 14 nM T76685 CF5C0L 46224950 IC50 = 18 nM T76685 CFEP51 46224951 IC50 = 19 nM T76685 C64XNW 46224952 IC50 = 55 nM T76685 CVP40Z 46224953 IC50 = 16 nM T76685 CU27FH 46224976 IC50 = 15 nM T76685 CR1GH2 46224977 IC50 = 0.41 nM T76685 CJ2IZ5 46224978 IC50 = 7.8 nM T76685 COK4N5 46224979 IC50 = 1.7 nM T76685 CW1C5J 46225007 IC50 = 5.8 nM T76685 CF0PT5 46225008 IC50 = 1.9 nM T76685 C8YS0O 46225009 IC50 = 7.5 nM T76685 C46PQM 46225010 IC50 = 71 nM T76685 C61FHM 46225032 IC50 = 0.49 nM T76685 C29WKZ 46225033 IC50 = 0.52 nM T76685 CSN5F6 46225034 IC50 = 1110 nM T76685 CXYU59 46225035 IC50 = 1.6 nM T76685 CT3W8V 46225067 IC50 = 2.2 nM T76685 C4IKY3 46225068 IC50 = 31 nM T76685 C6WU1H 46225069 IC50 = 1.2 nM T76685 C3SMQ7 46225070 IC50 = 7.3 nM T76685 CSWL98 46225106 IC50 = 4450 nM T76685 CT4Z3E 46225107 IC50 = 6250 nM T76685 CR16XN 46225108 IC50 = 13 nM T76685 C8HQ5L 46225109 IC50 = 1 nM T76685 CFD7G1 46225143 IC50 = 3.8 nM T76685 CHW67Q 46225144 IC50 = 9.2 nM T76685 COC30B 46225145 IC50 = 3 nM T76685 C8TV9Z 46225146 IC50 = 23 nM T76685 CB9X6O 46225186 IC50 = 5.7 nM T76685 C3JMV9 46225187 IC50 = 2.1 nM T76685 CB8XI0 46225188 IC50 = 5.7 nM T76685 C9GHP7 46225189 IC50 = 0.22 nM T76685 CT13RO 46225234 IC50 = 3.4 nM T76685 C6VA3F 46225235 IC50 = 27 nM T76685 CD7P8S 46225236 IC50 = 20 nM T76685 C6MYB5 46225237 IC50 = 17 nM T76685 CRSN07 46225286 IC50 = 199 nM T76685 CUD2J3 46225287 IC50 = 2.2 nM T76685 C1LN4P 46225288 IC50 = 2810 nM T76685 C5M9JO 46225289 IC50 = 2.1 nM T76685 C6D5UP 46226066 EC50 > 31622.78 nM T76685 C65MPA 46226067 EC50 > 31622.78 nM T76685 CC2Y3O 46226068 EC50 > 31622.78 nM T76685 CH9V2M 46226069 EC50 > 31622.78 nM T76685 C18GLZ 46226070 EC50 > 31622.78 nM T76685 CL0KM4 46226071 EC50 > 31622.78 nM T76685 C0T2WV 46226081 IC50 = 0.82 nM T76685 C4FC9X 46226082 IC50 = 0.4 nM T76685 C3UFW0 46226083 EC50 > 31622.78 nM T76685 C1Y2ZD 46226084 EC50 > 31622.78 nM T76685 C54MRO 46226085 EC50 > 31622.78 nM T76685 C97WVQ 46226086 EC50 > 31622.78 nM T76685 CXA8H5 46226087 EC50 > 31622.78 nM T76685 C3KQY6 46226088 Ki = 9900 nM T76685 CD07HW 46226089 Ki = 1615 nM T76685 C9M4EP 46226090 Ki > 10000 nM T76685 CZWU48 46226097 IC50 = 1.7 nM T76685 CBM21N 46226098 IC50 = 26 nM T76685 C4QCN5 46226099 IC50 = 51 nM T76685 C58RHI 46226108 EC50 > 31622.78 nM T76685 CR97PI 46226109 EC50 > 31622.78 nM T76685 C63IRS 46226110 EC50 = 3981.07 nM T76685 CAP1I4 46226111 EC50 > 31622.78 nM T76685 C64NOG 46226112 EC50 > 31622.78 nM T76685 CDH3B0 46226113 EC50 > 31622.78 nM T76685 CNV75F 46226114 Ki = 900 nM T76685 C4L2HM 46226115 Ki = 2500 nM T76685 CMDO26 46226116 Ki > 10000 nM T76685 C8GFT5 46226139 IC50 = 0.51 nM T76685 CDS2G6 46226147 EC50 > 31622.78 nM T76685 CVJF51 46226148 EC50 > 31622.78 nM T76685 CSI65H 46226149 EC50 = 19952.62 nM T76685 CWU43D 46226150 Ki = 2200 nM T76685 C1D3FQ 46226151 Ki = 2500 nM T76685 C6L4PR 46226152 Ki = 560 nM T76685 C8TG0B 46226158 IC50 = 0.54 nM T76685 CV7SD9 46226165 IC50 = 4.5 nM T76685 C0LK3O 46226166 IC50 = 5.8 nM T76685 CO1T7J 46226175 IC50 = 3.8 nM T76685 CS4FD7 46226231 IC50 = 0.3 nM T76685 C5WO0H 46226232 IC50 = 0.59 nM T76685 C1RYK4 46226233 IC50 = 21 nM T76685 C01LCN 46226249 IC50 = 1.1 nM T76685 C05TRK 46226268 IC50 = 0.79 nM T76685 CQ4H8C 46226270 IC50 = 3.7 nM T76685 C7KYV2 46226287 IC50 = 0.49 nM T76685 CV80ON 46226288 IC50 = 1.2 nM T76685 C4XOL6 46226289 IC50 = 0.11 nM T76685 C98TQN 46226305 IC50 = 0.11 nM T76685 C0DGW9 46226306 IC50 = 1.9 nM T76685 C5QMR4 46226307 IC50 = 5.5 nM T76685 CHC5P2 46226331 IC50 = 10 nM T76685 CT13UH 46226332 IC50 = 30 nM T76685 CSAC85 46226404 EC50 > 31622.78 nM T76685 CC5YA2 46226408 EC50 > 31622.78 nM T76685 CS79CQ 46226425 EC50 > 31622.78 nM T76685 CGWY69 46226426 EC50 > 31622.78 nM T76685 C5JDX0 46226427 EC50 > 31622.78 nM T76685 CA9NO8 46226428 EC50 = 2511.89 nM T76685 CR7K0F 46226429 EC50 = 6309.57 nM T76685 CXA5W9 46226430 EC50 > 31622.78 nM T76685 CEXZ31 46227715 Ki = 3100 nM T76685 CC29JS 46227721 Ki = 780 nM T76685 CV7H3L 46227722 Ki = 2500 nM T76685 C3OG7F 46227727 Ki = 830 nM T76685 CIH45R 46227729 Ki = 140 nM T76685 C67KXM 46227739 Ki = 1100 nM T76685 CPJ43K 46229257 Ki = 733 nM T76685 C34LAI 46229258 Ki > 10000 nM T76685 CTA7F0 46229282 Ki > 10000 nM T76685 CY7JA8 46229283 Ki > 10000 nM T76685 C6E5BK 46229284 Ki > 10000 nM T76685 C4GEX6 46229285 Ki = 2875 nM T76685 CIF9G1 46229732 Ki = 444 nM T76685 CNQ71K 46229733 Ki = 714 nM T76685 C6UFE7 46229734 Ki = 72 nM T76685 COG0D9 46229778 Ki > 1636 nM T76685 CEO0H4 46229779 Ki = 109 nM T76685 CW9NS3 46229780 Ki = 15 nM T76685 C8OCJ7 46229781 Ki = 467 nM T76685 C0H1NZ 46229782 Ki = 133 nM T76685 CTD56S 46229826 Ki = 63 nM T76685 CGEN85 46229827 Ki = 48 nM T76685 CQ9UG4 46229828 Ki = 158 nM T76685 CM2L5W 46229864 Ki = 6 nM T76685 CB5J0N 46229865 Ki = 2.3 nM T76685 CJ8YS5 46229866 Ki = 112 nM T76685 CR7CP6 46229896 Ki = 61 nM T76685 CF6P0K 46229897 Ki = 4.2 nM T76685 C7A9XG 46229898 Ki = 5.8 nM T76685 CWF2G6 46229969 Ki = 42 nM T76685 C5YE2W 46229970 Ki = 5.1 nM T76685 CV8O4J 46229971 Ki = 3.4 nM T76685 CI36WU 46230014 Ki = 8 nM T76685 C2TPH4 46230015 Ki = 554 nM T76685 C4FVX8 46230016 Ki = 690 nM T76685 C59CRV 46230017 Ki = 44 nM T76685 CV6KM4 46230070 Ki = 451 nM T76685 C6W3YJ 46230071 Ki = 13 nM T76685 CW3Z1X 46230072 Ki = 57 nM T76685 CSZ9L3 46230073 Ki = 33 nM T76685 CU7KB8 46230122 Ki = 18 nM T76685 C5ZC0J 46230123 Ki = 33 nM T76685 CDVT81 46230124 Ki = 35 nM T76685 C6J5SC 46230125 Ki = 16 nM T76685 C7Y3CB 46230705 IC50 = 28.2 nM T76685 C3UI7A 46230816 IC50 = 2.51 nM T76685 CDW1O9 46230974 Ki > 10000 nM T76685 CK31LV 46230975 Ki = 3995 nM T76685 C34LDI 46231031 Ki = 5444 nM T76685 CNW5V6 46231032 Ki = 1995 nM T76685 CB1OC6 46231088 Ki = 4152 nM T76685 C6FAH7 46231089 Ki > 10000 nM T76685 CL17TN 46231164 Ki > 1000 nM T76685 CWZ70O 46232373 Ki > 3000 nM T76685 CMZ9G4 46232374 Ki > 3000 nM T76685 C8E0NF 46232375 Ki > 3000 nM T76685 CKX9T8 46232376 Ki > 3000 nM T76685 C7SAY6 46232377 Ki > 3000 nM T76685 CP6D1J 46232431 Ki = 616 nM T76685 C6O8JZ 46232432 Ki = 1720 nM T76685 CZ1H6V 46232433 Ki > 3000 nM T76685 C9AOF0 46232434 Ki > 3000 nM T76685 CV02TB 46232435 Ki > 3000 nM T76685 CHE64C 46232505 Ki > 3000 nM T76685 CU36FE 46232506 Ki > 3000 nM T76685 C9UO1G 46232507 Ki > 3000 nM T76685 C30YXI 46232508 Ki > 3000 nM T76685 CZA8J2 46232547 Ki > 3000 nM T76685 CLI29U 46232548 Ki > 3000 nM T76685 CF8D6Z 46232549 Ki > 3000 nM T76685 CT02GZ 46232550 Ki > 3000 nM T76685 CC58RP 46232551 Ki > 3000 nM T76685 C3OYB9 46232577 Ki = 955 nM T76685 CNML95 46232578 Ki > 3000 nM T76685 CL0S8C 46232579 Ki = 0.24 nM T76685 C5Y8LD 46232580 Ki = 67.8 nM T76685 CCU94R 46232610 Ki = 11.7 nM T76685 CTYP68 46232611 Ki = 1340 nM T76685 C6QGB3 46232612 Ki = 333 nM T76685 COKU52 46232613 Ki > 3000 nM T76685 CS6UC7 46232638 Ki = 1840 nM T76685 CA94OK 46233073 Ki > 3000 nM T76685 C0VZ8J 46236057 Ki = 763 nM T76685 C6B5LZ 46239964 EC50 = 0.5 nM T76685 C5G3VL 46309339 Ki > 10000 nM T76685 C9IKL7 46833780 Ki > 1000 nM T76685 CSX30A 46834060 EC50 > 100000 nM T76685 CCT97N 46843358 EC50 > 50000 nM T76685 CNM5O6 46843431 EC50 > 50000 nM T76685 CV03HY 46843437 EC50 > 50000 nM T76685 C52SRT 46843872 EC50 > 20000 nM T76685 CN6M3Y 46851728 EC50 > 25000 nM T76685 C56HDV 46851886 EC50 > 25000 nM T76685 C43ZMW 46852048 EC50 > 25000 nM T76685 CK8N2W 46852211 EC50 > 25000 nM T76685 CD04SA 46852212 EC50 > 25000 nM T76685 CA9PE1 46852366 EC50 > 25000 nM T76685 C2QA8S 46856243 EC50 > 10000 nM T76685 C0J1EU 46856244 EC50 = 2550 nM T76685 CY3CE6 46861579 EC50 = 250 nM T76685 C97JEP 46871671 IC50 = 3 nM T76685 CFV3T7 46871949 EC50 = 96.9 nM T76685 CPAK05 46872381 EC50 > 20000 nM T76685 C95GAX 46872383 EC50 > 20000 nM T76685 C8INY3 46872497 EC50 = 5764 nM T76685 CK75SZ 46872613 EC50 > 20000 nM T76685 CQNL15 46873104 EC50 > 20000 nM T76685 CEZ42W 46873105 EC50 > 20000 nM T76685 C2F1LZ 46873202 EC50 > 20000 nM T76685 C6S2IH 46873203 EC50 = 1170 nM T76685 C6NK0P 46873310 EC50 > 20000 nM T76685 C02UDG 46873409 EC50 > 20000 nM T76685 CW0UE4 46873411 EC50 > 20000 nM T76685 CU95VF 46873412 EC50 = 217 nM T76685 CEX7G9 46873414 EC50 = 1965 nM T76685 CFYJ67 46873415 EC50 = 2940 nM T76685 CRU34K 46873515 EC50 > 20000 nM T76685 CV8F7U 46873516 EC50 = 13000 nM T76685 C4DQ0A 46880367 Ki = 84 nM T76685 C6OE4K 46880408 Ki = 21.7 nM T76685 CSE86Q 46880409 Ki = 53 nM T76685 C2A3WU 46880410 Ki = 37 nM T76685 C4GQH2 46880411 Ki = 11.3 nM T76685 C6X7SW 46880499 Ki = 58 nM T76685 C9XJ0K 46880500 Ki = 280 nM T76685 C6N8WX 46880632 Ki = 463 nM T76685 CK3WD5 46880678 Ki > 1000 nM T76685 CKH6J7 46884054 IC50 = 13 nM T76685 CVY2T4 46888365 IC50 = 2 nM T76685 CO7M5J 46888366 IC50 = 0.6 nM T76685 CLS1G3 46888367 IC50 = 0.6 nM T76685 CGD6T5 46888386 IC50 = 1.3 nM T76685 C13SVO 46888387 IC50 = 1.2 nM T76685 C9G2HI 46888388 IC50 = 56 nM T76685 C5D2CK 46888389 IC50 = 1.1 nM T76685 CME5D6 46888413 IC50 = 480 nM T76685 CV0JO1 46888438 IC50 = 7.65 nM T76685 CDUM26 46888645 IC50 = 6.5 nM T76685 CTN16E 46888688 IC50 = 0.7 nM T76685 C4SX5W 46888719 IC50 = 0.6 nM T76685 CT8E9F 46888720 IC50 = 4 nM T76685 CP75RD 46888721 IC50 = 1.3 nM T76685 C9Z2CO 46888748 IC50 = 2.1 nM T76685 CR7HN9 46888749 IC50 = 0.2 nM T76685 C06HUF 46888750 IC50 = 0.5 nM T76685 CEMZ98 46888775 IC50 = 1.4 nM T76685 CYT7P0 46888776 IC50 = 0.2 nM T76685 CJDH10 46888777 IC50 = 0.3 nM T76685 CM6S8Z 46888778 IC50 = 0.2 nM T76685 C7R9KO 46889225 Ki = 12 nM T76685 C9R0CB 46890855 IC50 = 21 nM T76685 CN5E1A 46890915 IC50 = 1.7 nM T76685 C6OSC8 46890967 IC50 = 790 nM T76685 CA2V8W 46891079 IC50 = 80 nM T76685 COQ1S6 46891146 IC50 = 19 nM T76685 C7T2GX 46909057 IC50 = 30000 nM T76685 C2A7QJ 46911281 IC50 = 1.4 nM T76685 CL47EI 46911790 Ki = 11.6 nM T76685 C8YLX7 46912919 Ki = 1 nM T76685 CD31GS 46914568 Ki = 2080 nM T76685 CCDY16 46914722 Ki > 10000 nM T76685 C43TQI 46914723 Ki = 460 nM T76685 CZS28Q 46914724 Ki > 10000 nM T76685 C1PK8H 46914725 Ki > 10000 nM T76685 CD1T3Z 46914726 Ki > 10000 nM T76685 CIG17Z 46914868 Ki > 10000 nM T76685 CMV18T 46914869 Ki > 10000 nM T76685 CXGF68 46914870 Ki > 10000 nM T76685 C10IJF 46914871 Ki > 10000 nM T76685 C5US1J 46915018 Ki > 10000 nM T76685 C72YRK 46915019 Ki > 10000 nM T76685 C48PXG 46915021 Ki > 10000 nM T76685 C08DTP 46915022 Ki > 10000 nM T76685 C4TXE9 46915181 Ki = 510 nM T76685 C3ZLI4 46915182 Ki = 360 nM T76685 C2HQ5I 46915183 Ki = 245.7 nM T76685 C5T4EW 46915184 Ki > 10000 nM T76685 C9ZMB6 46915338 Ki > 10000 nM T76685 CK36UG 46915339 Ki > 10000 nM T76685 C15YSX 46915340 Ki > 10000 nM T76685 CT1P4V 46915341 Ki > 10000 nM T76685 CIDJ51 46915342 Ki = 29.7 nM T76685 C24CMT 46915484 Ki > 10000 nM T76685 CP3T2G 46915629 Ki > 10000 nM T76685 C3L2BF 46915632 Ki = 900 nM T76685 CR1K7X 46915633 Ki > 10000 nM T76685 CN0A1F 46915770 Ki = 3210 nM T76685 CHG94W 46915775 Ki > 10000 nM T76685 C90CHW 46915915 Ki > 10000 nM T76685 CIO5Y8 46916568 Ki = 6000 nM T76685 CZ4PY1 46919791 Ki = 12.59 nM T76685 CJ70AD 46919792 Ki = 1.995 nM T76685 C3K0LS 46934582 IC50 = 5 nM T76685 CT8Z7B 48127247 Ki = 56 nM T76685 CS4LC8 48131648 Ki = 800 nM T76685 CWEH82 48134599 Ki = 386 nM T76685 CN4Q7O 49779469 Ki > 3000 nM T76685 CPW56Y 49780575 Ki = 94 nM T76685 CB68TP 49780791 Ki = 41.9 nM T76685 C2B6NH 49780792 Ki = 30.4 nM T76685 CNCG41 49780793 Ki = 4.41 nM T76685 CO7W4M 49781019 EC50 = 27.9 nM T76685 C3B1WZ 49781020 Ki = 37 nM T76685 C4OJ3P 49781021 Ki = 6.35 nM T76685 CKE6A5 49781237 Ki = 17.3 nM T76685 CZ7M0W 49781238 Ki = 94.1 nM T76685 CB91JD 49781239 Ki = 1292 nM T76685 C9I2YR 49781454 Ki = 506 nM T76685 C1NLT8 49781455 Ki > 2500 nM T76685 CB24YU 49781456 Ki = 230 nM T76685 CR4KL0 49781457 Ki = 19.5 nM T76685 CNW96U 49781458 Ki = 5.44 nM T76685 C2DWZ4 49781682 Ki = 2.3 nM T76685 CAD7R3 49781683 Ki = 88.8 nM T76685 CCW7S8 49781684 Ki = 15.5 nM T76685 C35OZF 49781685 Ki = 6.12 nM T76685 CXPZ67 49781896 Ki = 5.51 nM T76685 CM8CT6 49819854 Ki > 3000 nM T76685 CAP20Y 49819855 Ki > 1000 nM T76685 C2H3LB 49819856 Ki = 626 nM T76685 CY54HV 49820008 Ki > 3000 nM T76685 C1XHJ3 49820009 Ki = 592 nM T76685 C1I6ES 49820010 Ki = 596 nM T76685 C1UBA0 49820012 Ki > 1000 nM T76685 CM93PJ 49820013 Ki = 929 nM T76685 CC91QZ 49820163 Ki = 131 nM T76685 C45VYH 49820164 Ki > 1000 nM T76685 CZX25W 49820165 Ki > 3000 nM T76685 CAU16J 49820166 Ki > 1000 nM T76685 CQ78GC 49820167 Ki = 454 nM T76685 CI26US 49820318 Ki > 1000 nM T76685 C5SYJ4 49820319 Ki > 1000 nM T76685 CHI43J 49820320 Ki > 1000 nM T76685 CS94OJ 49820321 Ki = 562 nM T76685 CM9E4A 49820322 Ki = 548 nM T76685 CU0P1L 49820323 Ki > 1000 nM T76685 CQCN46 49820469 Ki > 1000 nM T76685 C1UGS6 49820621 Ki > 1000 nM T76685 C7ZY1V 49820624 Ki = 105.1 nM T76685 CH73VZ 49820626 Ki = 193.4 nM T76685 C1UR2D 49820779 Ki > 1000 nM T76685 CG9H5Z 49820783 Ki > 3000 nM T76685 C0GD7O 49820784 Ki > 1000 nM T76685 CYG4A0 49824032 Ki = 34673.69 nM T76685 C7MR2D 49840760 Ki > 3000 nM T76685 CN89JQ 49840830 Ki > 1000 nM T76685 C6QS1A 49840831 Ki = 51.2 nM T76685 CFK8J2 49840832 Ki = 34.4 nM T76685 CM0D5J 49840833 Ki = 134 nM T76685 CRV02J 49840834 Ki = 384 nM T76685 CC05PM 49840907 Ki > 1000 nM T76685 C9JE6I 49840908 Ki > 1000 nM T76685 CXI14S 49840909 Ki > 3000 nM T76685 CR5M8V 49840911 Ki > 3000 nM T76685 CTH8K1 49843511 Ki = 0.12 nM T76685 C9K1PB 49847679 EC50 = 1400 nM T76685 CZK27C 49848443 EC50 > 50000 nM T76685 C32PJB 49855337 EC50 = 0.631 nM T76685 CQZB40 49861285 Ki > 10000 nM T76685 CB3DX7 49862509 EC50 = 31.62 nM T76685 CD03BK 49862563 EC50 = 25.12 nM T76685 CA24NE 49862564 EC50 > 10000 nM T76685 CS8GW5 49862565 EC50 = 158.49 nM T76685 CICK43 49862566 EC50 = 100 nM T76685 CD2TR6 49862582 IC50 = 22 nM T76685 CJB8M0 49862583 IC50 = 340 nM T76685 CV06BA 49862615 EC50 = 3981.07 nM T76685 CJ95AK 49862616 EC50 = 3.981 nM T76685 CU5H3T 49862617 EC50 = 125.89 nM T76685 C67MVR 49862639 IC50 = 1300 nM T76685 CG2L3T 49862640 IC50 = 810 nM T76685 CWJ2C0 49862666 Ki = 1.259 nM T76685 CWR02I 49862667 EC50 = 501.19 nM T76685 C3GL7S 49862668 EC50 = 63.1 nM T76685 C8E0NZ 49862701 IC50 = 2000 nM T76685 C1XC4V 49862753 EC50 = 794.33 nM T76685 CSH8C5 49862754 EC50 = 6.31 nM T76685 CSCJ63 49862755 EC50 = 5.012 nM T76685 CV47MH 49864283 Ki = 2.8 nM T76685 C9UAP2 49864284 Ki = 1900 nM T76685 CKZ76J 49864285 Ki = 1700 nM T76685 C7Y9FB 49864287 Ki = 480 nM T76685 C7Y1GV 49865614 Ki = 52 nM T76685 CHC10N 49865615 Ki = 15.3 nM T76685 CSGK87 49865616 Ki = 11.9 nM T76685 CD0CJ2 49865617 Ki = 33.1 nM T76685 CTC3W1 49865618 Ki = 70 nM T76685 C1VUG0 49865655 EC50 = 31.62 nM T76685 C7AWN5 49865656 EC50 = 7.943 nM T76685 CN83QV 49865683 Ki = 16.1 nM T76685 C2JX4A 49865713 EC50 = 3.981 nM T76685 C74RSL 49866076 IC50 = 104 nM T76685 CD74FG 49866077 IC50 = 64 nM T76685 CBL30H 49866078 IC50 = 269 nM T76685 CUP89G 49866079 IC50 = 21 nM T76685 C3N4QT 49866144 IC50 = 73 nM T76685 CB8QE6 49866145 IC50 = 51 nM T76685 CHDZ51 49866146 IC50 = 58 nM T76685 CO21VX 49866147 IC50 = 37 nM T76685 CX8UP9 49866182 IC50 = 45 nM T76685 C6YJ2V 49866183 IC50 = 7 nM T76685 CMI8U1 49866184 IC50 = 45 nM T76685 C7R2YS 49866185 IC50 = 3 nM T76685 C5GOP7 49866224 IC50 = 23 nM T76685 C56PIQ 49866225 IC50 = 7 nM T76685 CR3F0V 49866226 IC50 = 27 nM T76685 C8Y9CP 49866230 Ki = 15.6 nM T76685 CGS8V1 49866249 IC50 = 19 nM T76685 CS7TP4 49866255 Ki = 16.1 nM T76685 C0BQ4U 49890666 Ki = 5040 nM T76685 C2RY0J 50878551 Ki > 10000 nM T76685 CKBS87 50898695 Ki > 10000 nM T76685 CFA38L 50898696 Ki > 10000 nM T76685 CP46YL 50898697 Ki > 10000 nM T76685 C3PIV5 50898698 Ki > 10000 nM T76685 C3B0HL 50907287 Ki = 550.3 nM T76685 CNM78T 50907288 Ki = 272.6 nM T76685 C7AVR3 50907289 Ki = 81 nM T76685 C0RGF2 50907490 Ki = 534.4 nM T76685 CGHI15 50907491 Ki = 124.1 nM T76685 C13OJL 50907492 Ki = 211 nM T76685 CMT0K4 50907493 Ki = 290.1 nM T76685 CHAB52 50907494 Ki = 123.1 nM T76685 CC0B4J 50907495 Ki = 182.1 nM T76685 C20WYJ 50907705 Ki = 372.3 nM T76685 C9H8UP 50907706 Ki = 311.4 nM T76685 CB7V4R 50907707 Ki = 97.2 nM T76685 C7R5KQ 50907708 Ki = 368.2 nM T76685 C2X9WV 50907709 Ki = 518.9 nM T76685 C0MZA9 50907710 Ki = 89.5 nM T76685 C6RF7I 50907920 Ki = 47.6 nM T76685 CW39DE 50907921 Ki = 45.6 nM T76685 COCB87 50907922 Ki = 157.5 nM T76685 CM7W3P 50907923 Ki = 233.5 nM T76685 CK6MT8 50907924 Ki = 150.7 nM T76685 C1S4IB 50907925 Ki = 193.5 nM T76685 CS8MX3 50908151 Ki = 37.5 nM T76685 CT0IA2 50908152 Ki = 104.7 nM T76685 CVC8L6 50908153 Ki = 90.7 nM T76685 C1YF6I 50915132 EC50 > 10000 nM T76685 CC0DR4 50941835 EC50 > 10000 nM T76685 C9WA0L 51029725 EC50 > 10000 nM T76685 C2IH9K 51030930 EC50 > 10000 nM T76685 CX4PF6 51030931 EC50 > 10000 nM T76685 C31UWX 51042138 Ki > 10000 nM T76685 CAO41L 51351511 EC50 > 20000 nM T76685 C9AZ3J 51357040 Ki = 2400 nM T76685 C8T1BE 51357043 Ki = 1600 nM T76685 C3BRM2 51357044 Ki > 10000 nM T76685 CIZ96K 51357316 Ki = 1300 nM T76685 C5RXF2 51357319 Ki = 1380 nM T76685 C6G9SM 51357595 Ki = 600 nM T76685 C1R0DP 51357597 Ki = 1700 nM T76685 CU0I5S 51357598 Ki > 40000 nM T76685 CE3H6X 51357599 Ki > 40000 nM T76685 CGV79B 51357600 Ki = 800 nM T76685 C6S1KB 51357868 Ki = 4000 nM T76685 CD9FL1 52918122 IC50 > 17000 nM T76685 CRWO47 52918123 IC50 > 17000 nM T76685 CC2O0K 52918124 IC50 = 5020 nM T76685 CHR92P 52941287 EC50 = 501.19 nM T76685 CY54QP 52941289 EC50 = 1000 nM T76685 C0HQV7 52941294 EC50 = 316.23 nM T76685 CA1F9R 52941334 EC50 = 1995.26 nM T76685 C69TMB 52941604 Ki > 10000 nM T76685 C54BIX 52943703 EC50 = 100 nM T76685 CG9A2Y 52943719 Ki > 10000 nM T76685 CD4MK9 52943735 EC50 = 158.49 nM T76685 CE7K2D 52944154 IC50 = 0.3 nM T76685 C5B7KN 52944375 Ki > 10000 nM T76685 C53SIC 52944884 EC50 = 100 nM T76685 CZS26J 52944885 EC50 = 12.59 nM T76685 CL0IT3 52944886 Ki > 10000 nM T76685 C46GIZ 52944912 Ki > 10000 nM T76685 CN9P8H 52944915 EC50 = 630.96 nM T76685 CADT74 52944916 EC50 = 100 nM T76685 CX85GV 52946094 EC50 = 19.95 nM T76685 CUL1B5 52946095 Ki > 10000 nM T76685 CVC06D 52946132 EC50 > 10000 nM T76685 C8ZY4U 52946150 EC50 = 31.62 nM T76685 CEC42Q 52947367 EC50 = 63.1 nM T76685 CB2LF5 52947371 Ki > 10000 nM T76685 CQWZ29 52947376 Ki > 10000 nM T76685 C87AFQ 52947385 Ki > 10000 nM T76685 CC9Q1I 52947697 Ki > 10000 nM T76685 C5H7EL 52948053 Ki > 10000 nM T76685 CT0XY2 52948592 Ki > 10000 nM T76685 CN16UM 52948595 Ki > 10000 nM T76685 C3KGT9 52949778 EC50 = 63.1 nM T76685 C09DXM 52949805 Ki > 10000 nM T76685 C1LSQ4 52949819 EC50 = 1258.93 nM T76685 C9ADM3 52950114 Ki > 10000 nM T76685 C9C1FN 52951268 Ki = 297 nM T76685 CXF3Z8 52951269 Ki > 10000 nM T76685 C6AVI3 52951270 Ki > 10000 nM T76685 C5DRM0 52951271 Ki > 10000 nM T76685 C1LD4S 52951378 Ki > 10000 nM T76685 C8OMI5 52951379 Ki > 10000 nM T76685 CI47GU 52951380 Ki = 437 nM T76685 CM0D9Z 52951381 Ki > 10000 nM T76685 CV1BX8 52951382 Ki = 259 nM T76685 CLY37M 52951383 Ki > 10000 nM T76685 CC63FQ 52951479 Ki = 500 nM T76685 C06YFP 52951480 Ki = 115 nM T76685 CPA2G4 52951481 Ki = 62.2 nM T76685 CYP0I3 52951482 Ki = 15.7 nM T76685 CAF5K3 52951483 Ki = 680 nM T76685 CZC4B0 52951484 Ki > 10000 nM T76685 CI5M7G 52951606 Ki = 356 nM T76685 CN39RI 52951607 Ki = 55 nM T76685 C51UGF 52951608 Ki > 10000 nM T76685 C7VN2Z 53249197 Ki = 17.2 nM T76685 CJXH50 53316569 Ki > 3000 nM T76685 CH5J7F 53316956 EC50 = 251.19 nM T76685 CB5F8M 53316957 EC50 = 199.53 nM T76685 CWCA05 53316975 Ki = 42 nM T76685 C8S0EL 53317367 EC50 = 8500 nM T76685 C7M9BI 53317422 EC50 > 1000 nM T76685 CS8C4D 53317423 EC50 = 1294 nM T76685 C9XJ4D 53317638 Ki = 1800 nM T76685 C8P2MZ 53318246 EC50 = 794.33 nM T76685 CDZ2R3 53318301 Ki = 2100 nM T76685 CT8OS9 53318302 Ki = 130 nM T76685 C4GL7O 53318303 Ki = 5444 nM T76685 CW6J9C 53318654 EC50 = 2450 nM T76685 C7IH8G 53318655 EC50 = 25 nM T76685 CQSZ57 53318656 EC50 = 320 nM T76685 CF1BS7 53318713 EC50 > 10000 nM T76685 CHC3R5 53319210 Ki = 368 nM T76685 CRO12M 53319609 EC50 = 199.53 nM T76685 CJ0M5I 53319626 Ki = 95 nM T76685 C6V5OU 53319661 Ki > 10000 nM T76685 C8R6XB 53319972 EC50 = 12550 nM T76685 CW8EQ3 53320023 EC50 = 130 nM T76685 CRS79K 53320272 EC50 > 10000 nM T76685 CI80DM 53320925 Ki = 1700 nM T76685 C4VAP1 53321340 EC50 > 1000 nM T76685 CJ7TL9 53322235 EC50 = 15.85 nM T76685 CJQT01 53322236 EC50 = 79.43 nM T76685 CJE6F1 53322251 Ki = 28 nM T76685 CBD23U 53322256 Ki = 480 nM T76685 CFQY21 53322288 Ki = 1422 nM T76685 CZA30O 53322289 Ki = 53 nM T76685 CVP47L 53322598 EC50 = 39 nM T76685 C8JLS1 53322599 EC50 > 10000 nM T76685 CY9ZK2 53322600 EC50 > 10000 nM T76685 C5USQ2 53323572 EC50 = 158.49 nM T76685 CZ60KM 53323573 EC50 = 31.62 nM T76685 CO7ED9 53323994 EC50 > 1000 nM T76685 CNJQ28 53323995 EC50 > 1000 nM T76685 CP8CN3 53323996 EC50 = 2290 nM T76685 CS9I8F 53323997 EC50 = 665 nM T76685 CNMF87 53324282 EC50 = 1055 nM T76685 CO9IA6 53324879 EC50 = 398.11 nM T76685 C31DKS 53324880 EC50 = 79.43 nM T76685 CO7BF5 53324934 Ki = 1100 nM T76685 CN6VT3 53324935 Ki = 650 nM T76685 CQ7ME2 53325220 EC50 = 140 nM T76685 CF2DQ0 53325221 EC50 = 1800 nM T76685 C6T9OP 53325289 EC50 > 1000 nM T76685 CFCT05 53325377 EC50 = 3250 nM T76685 C4IF0H 53326153 EC50 = 15.85 nM T76685 C2T8ED 53326154 EC50 = 100 nM T76685 CD2P3Z 53326155 EC50 = 1995.26 nM T76685 C2VR6O 53326220 Ki = 4100 nM T76685 C4BLU0 53326382 EC50 = 79.43 nM T76685 CW7PM5 53326510 EC50 = 87 nM T76685 C1ZF7K 53326560 EC50 > 1000 nM T76685 CK3I2Y 53353783 Ki = 7410 nM T76685 CSQM04 53356799 Ki = 65 nM T76685 CYG6Q1 53358318 EC50 > 10 nM T76685 C5ZHE4 53377393 Ki = 0.67 nM T76685 C3X7OW 53386375 EC50 > 100000 nM T76685 CW91SC 53387189 Ki > 10000 nM T76685 CKSB51 53387350 Ki > 10000 nM T76685 CKE02W 53387351 Ki = 31.3 nM T76685 CH37DN 53387419 Ki > 2000 nM T76685 CFJG62 53387420 Ki = 2000 nM T76685 C7HRK8 53387421 Ki = 2000 nM T76685 CQZF69 53387584 Ki = 2000 nM T76685 CM47GI 53387585 Ki = 2000 nM T76685 CQ81LN 53387586 Ki > 5000 nM T76685 CN67QX 53387587 Ki = 221 nM T76685 C0GI9B 53387746 Ki = 84.7 nM T76685 CS8B2H 53392078 Ki = 689 nM T76685 C6RKL5 53392169 Ki > 10000 nM T76685 CM8T0J 53392248 Ki = 200 nM T76685 CGZD15 53392250 Ki > 10000 nM T76685 CZ18IO 53392334 Ki > 10000 nM T76685 CE29LJ 53392335 Ki > 10000 nM T76685 CLBE83 53392336 Ki > 10000 nM T76685 CPKH67 53394451 Ki > 10000 nM T76685 CYQ7H1 53394457 Ki > 10000 nM T76685 CV5NQ4 53476894 EC50 > 100000 nM T76685 C6VLZ9 53483967 Ki = 8 nM T76685 CUBX46 53483982 Ki = 15 nM T76685 C2TP3Z 53494923 Ki > 10000 nM T76685 CP8MN1 53494924 Ki > 10000 nM T76685 CG9L7V 53494925 Ki > 10000 nM T76685 CO1K2X 53494926 Ki > 10000 nM T76685 CR4N3X 54577602 Ki = 163400 nM T76685 CX91HL 54579950 EC50 > 20000 nM T76685 C7I3ZC 54579951 EC50 > 20000 nM T76685 CGR29V 54580011 IC50 = 199 nM T76685 C1HC5S 54580064 EC50 = 5.012 nM T76685 CQ8AZ0 54580065 EC50 = 630.96 nM T76685 CYM8N2 54580066 EC50 = 79.43 nM T76685 CT2FB8 54580068 EC50 = 39.81 nM T76685 C4KGT2 54580069 EC50 = 63.1 nM T76685 CL5V4H 54580071 EC50 = 1.995 nM T76685 C3SER0 54580114 IC50 = 0.631 nM T76685 CX4ED5 54580115 IC50 = 2.57 nM T76685 C0E3DA 54580116 IC50 = 4.898 nM T76685 CG84FC 54580117 IC50 = 8.913 nM T76685 CDO2B0 54580174 IC50 = 12700 nM T76685 CS2PI0 54580175 IC50 > 17000 nM T76685 C5N2YX 54580194 IC50 = 930 nM T76685 C5AVO4 54580197 IC50 = 2022 nM T76685 CZG6L5 54580223 IC50 > 17000 nM T76685 CB37OP 54580227 IC50 = 3441 nM T76685 CVU32Y 54580228 IC50 = 1002 nM T76685 CFE51I 54580229 IC50 > 17000 nM T76685 C4VGN2 54580230 IC50 > 17000 nM T76685 C9G0UX 54580231 IC50 = 4044 nM T76685 CKLR94 54580466 EC50 > 20000 nM T76685 CSR9V2 54580931 EC50 > 20000 nM T76685 CZH49F 54581047 IC50 = 5.37 nM T76685 C4GAB9 54581050 EC50 = 251.19 nM T76685 CP7HC3 54581052 EC50 = 50.12 nM T76685 CV3SW1 54581091 IC50 = 0.5129 nM T76685 C19GPR 54581092 IC50 = 1.479 nM T76685 C5SK4C 54581093 IC50 = 2.63 nM T76685 C9YD6K 54581168 IC50 = 705 nM T76685 C72HZB 54581169 IC50 > 17000 nM T76685 C43FAB 54581198 IC50 > 17000 nM T76685 C9FO1C 54581199 IC50 = 188 nM T76685 C4P8NW 54581223 IC50 = 261 nM T76685 C4AE7R 54581224 IC50 > 17000 nM T76685 CUC36A 54581225 IC50 > 17000 nM T76685 CVK59Q 54581226 IC50 > 17000 nM T76685 C7ZL8M 54581476 EC50 > 20000 nM T76685 C8K7RL 54581988 EC50 > 20000 nM T76685 C6FU2I 54581989 EC50 > 20000 nM T76685 CG10LW 54582092 EC50 = 3.981 nM T76685 CL52TN 54582094 EC50 = 2.512 nM T76685 CB6DW8 54582096 EC50 = 10 nM T76685 CF9C2B 54582132 IC50 = 6.026 nM T76685 CZ1NQ0 54582133 IC50 = 9.333 nM T76685 CF39HJ 54582173 IC50 = 90 nM T76685 C3T7CY 54582249 IC50 > 17000 nM T76685 CJX1K9 54582251 IC50 > 17000 nM T76685 C3GM8O 54582252 IC50 > 17000 nM T76685 CP64NQ 54582479 EC50 > 20000 nM T76685 C5PZ4A 54582480 EC50 = 20000 nM T76685 CG3FA5 54582481 EC50 > 20000 nM T76685 CFG5J2 54582482 EC50 > 20000 nM T76685 C61IJU 54582925 EC50 > 20000 nM T76685 CPHS82 54582991 IC50 = 141 nM T76685 CP8TG1 54583028 EC50 = 63.1 nM T76685 CHT78R 54583030 EC50 = 6.31 nM T76685 C3QG4F 54583077 Ki = 5.495 nM T76685 CX3RS2 54583078 Ki = 5.012 nM T76685 CJ0F2K 54583160 IC50 > 17000 nM T76685 C08ONK 54583196 IC50 > 17000 nM T76685 CCS50N 54583230 IC50 > 17000 nM T76685 C0ET3G 54583455 EC50 > 20000 nM T76685 CD2BN6 54583456 EC50 > 20000 nM T76685 CDF83A 54583457 EC50 > 20000 nM T76685 C4G9CW 54583926 EC50 > 20000 nM T76685 C06IDY 54583927 EC50 > 20000 nM T76685 CEFL09 54584078 IC50 = 0.5754 nM T76685 CF76UY 54584079 IC50 = 1.549 nM T76685 C3TLJ2 54584080 IC50 = 5.129 nM T76685 CNQC76 54584153 IC50 > 17000 nM T76685 CJZS79 54584190 IC50 = 1528 nM T76685 C0K9SP 54584191 IC50 > 17000 nM T76685 CX2EJ4 54584192 IC50 > 17000 nM T76685 C8THZ7 54584193 IC50 > 17000 nM T76685 CXZL01 54584423 EC50 > 20000 nM T76685 CNVG29 54584424 EC50 > 20000 nM T76685 CFJ1G3 54584425 EC50 > 20000 nM T76685 C37TZQ 54584868 EC50 > 20000 nM T76685 C3FQE0 54584985 IC50 = 5.129 nM T76685 C8P6MI 54584991 EC50 = 79.43 nM T76685 C1B0TX 54585026 IC50 = 1.318 nM T76685 C9FJ2V 54585027 IC50 = 1.479 nM T76685 C4EB1D 54585060 IC50 = 2229 nM T76685 COQ86B 54585087 IC50 = 347 nM T76685 CVG86Q 54585088 IC50 = 68 nM T76685 CA7ZM4 54585089 IC50 > 17000 nM T76685 CV6PE4 54585090 IC50 > 17000 nM T76685 C0B6DK 54585147 IC50 > 17000 nM T76685 CK9N2B 54585148 IC50 > 17000 nM T76685 C47CQF 54585149 IC50 > 17000 nM T76685 C30LYP 54585371 EC50 = 25.12 nM T76685 C7TF3G 54585381 EC50 = 19300 nM T76685 C19LYO 54585382 EC50 = 19800 nM T76685 C3CIW8 54585835 EC50 > 20000 nM T76685 C60ZBV 54585836 EC50 > 20000 nM T76685 CUI9N5 54585837 EC50 > 20000 nM T76685 C8OR2E 54585941 EC50 = 50.12 nM T76685 CJLB09 54586104 IC50 > 17000 nM T76685 CY7XN2 54586105 IC50 = 4247 nM T76685 C78MRT 54586106 IC50 > 17000 nM T76685 CQ74VR 54586107 IC50 = 3445 nM T76685 CYCN52 54586108 IC50 > 17000 nM T76685 CE7WF1 54586109 IC50 > 17000 nM T76685 CNHM97 54586338 EC50 > 20000 nM T76685 CM14QB 54586803 EC50 > 20000 nM T76685 CG56XR 54586804 EC50 > 20000 nM T76685 CQWI92 54586805 EC50 > 20000 nM T76685 C4L5SW 54586806 EC50 > 20000 nM T76685 C5RKS0 54586916 IC50 = 8.318 nM T76685 C59FXV 54586919 EC50 = 15.85 nM T76685 CTK5S1 54586921 EC50 = 398.11 nM T76685 CW53CF 54586964 Ki = 7.586 nM T76685 C3PUX8 54586965 IC50 = 8.128 nM T76685 CMF92B 54587073 IC50 = 963 nM T76685 CM6Q8R 54587074 IC50 > 17000 nM T76685 CK6Q9F 54587075 IC50 = 312 nM T76685 CA37WI 54587108 IC50 > 17000 nM T76685 CZ23AJ 54587109 IC50 > 17000 nM T76685 CT8GH6 54587110 IC50 > 17000 nM T76685 CBI84E 54587111 IC50 > 17000 nM T76685 CCOF62 54587112 IC50 > 17000 nM T76685 C4XT9S 54587370 EC50 > 20000 nM T76685 C4GJ1Z 54587371 EC50 > 20000 nM T76685 CB49IH 54587372 EC50 > 20000 nM T76685 C1Q5RX 54587373 EC50 > 20000 nM T76685 C6H9US 54592384 Ki = 13 nM T76685 CUV69N 54669855 Ki = 750 nM T76685 CU9W8M 54680181 Ki > 1000 nM T76685 CDR58P 54732041 Ki > 10000 nM T76685 CJON78 54732042 Ki = 270 nM T76685 CE61UL 54752945 Ki = 1.259 nM T76685 CW28JF 54752946 Ki = 12.59 nM T76685 C3P9HQ 54752947 Ki > 1000 nM T76685 CG16QF 54769828 Ki > 10000 nM T76685 C8G2CW 54769829 Ki = 62 nM T76685 CU09YW 54769830 Ki > 10000 nM T76685 C8IH2D 56597771 Ki = 1300 nM T76685 CQ69YX 56599474 IC50 > 10000 nM T76685 CX8BT4 56642292 Ki = 31.62 nM T76685 C23NFV 56642293 Ki = 7.943 nM T76685 CU9D7V 56642294 Ki = 6.31 nM T76685 C9X8UN 56642295 Ki > 1000 nM T76685 C26KYO 56642422 Ki = 251.19 nM T76685 C8SXT3 56642423 Ki = 251.19 nM T76685 C0A5ML 56642424 Ki = 63.1 nM T76685 C3AC0D 56642425 Ki > 1000 nM T76685 CD8EG3 56642426 Ki > 1000 nM T76685 CW4V3C 56642427 Ki = 501.19 nM T76685 CZ7O2R 56642428 EC50 = 100 nM T76685 CE2B6T 56642541 EC50 = 50.12 nM T76685 CS6MJ7 56658151 Ki = 26 nM T76685 CFN58G 56659453 Ki = 82 nM T76685 C25NUZ 56659454 Ki = 0.81 nM T76685 C7V3XG 56659455 Ki = 27 nM T76685 CX1YD2 56659487 Ki = 8.2 nM T76685 CO30WQ 56659488 Ki = 0.37 nM T76685 CB6K8P 56659489 Ki = 0.2 nM T76685 C8F2LW 56661658 Ki = 61 nM T76685 CKLR96 56661659 Ki = 786 nM T76685 CI2E6F 56661776 Ki = 20 nM T76685 C5B2WH 56662770 Ki > 10000 nM T76685 CWS52M 56662852 Ki > 19400 nM T76685 CPSB19 56662902 Ki = 19 nM T76685 CV7SJ3 56662947 Ki = 1.4 nM T76685 CZXH42 56666243 Ki > 10000 nM T76685 C0J2LE 56666384 Ki = 21 nM T76685 CACK59 56666385 Ki = 10 nM T76685 CU57MG 56666387 Ki = 11 nM T76685 CME9V1 56666420 Ki = 0.18 nM T76685 CNWQ23 56668510 Ki = 260 nM T76685 CA3ZL8 56668680 Ki = 60 nM T76685 CRV05W 56669650 Ki = 5055 nM T76685 CAX2K8 56669651 Ki = 864000 nM T76685 C6R9VZ 56669796 Ki = 1.3 nM T76685 CHLT70 56669797 Ki = 335 nM T76685 CVF45I 56669798 Ki = 0.29 nM T76685 CEV08M 56669837 Ki = 1.5 nM T76685 C5FW7K 56669838 Ki = 0.47 nM T76685 CU83EN 56669839 Ki = 0.52 nM T76685 CA3V1W 56673163 Ki > 10000 nM T76685 C5U3AW 56673292 Ki = 1.2 nM T76685 C7SE6V 56673308 Ki = 11 nM T76685 CI6YQ2 56673320 Ki = 0.49 nM T76685 CK64EV 56675389 Ki > 10000 nM T76685 C17MNC 56676487 Ki > 10000 nM T76685 C8L9MT 56676610 Ki = 2.4 nM T76685 C4B7KC 56676611 Ki = 0.54 nM T76685 C9U5XM 56676663 Ki = 0.71 nM T76685 CBM0X1 56679803 Ki > 10000 nM T76685 C7V8DA 56679805 Ki = 2398000 nM T76685 C03JXE 56679953 Ki = 33 nM T76685 CZKU76 56679954 Ki = 610 nM T76685 CA60DY 56679955 Ki = 510 nM T76685 CLQ0O1 56683134 Ki > 10000 nM T76685 C30ADJ 56683280 Ki = 220 nM T76685 CA2Q9L 56683319 Ki = 0.38 nM T76685 C0GYJ1 56683320 Ki = 0.3 nM T76685 CV0S7J 56683321 Ki = 0.65 nM T76685 CO3WT8 56683322 Ki = 16.5 nM T76685 C2MFV5 56835155 EC50 > 10000 nM T76685 CP4WL5 56835156 EC50 = 3428 nM T76685 C78GIO 56835165 Ki = 10 nM T76685 CWE8D9 56837837 Ki = 2.3 nM T76685 C6B1MZ 56837838 Ki = 15.3 nM T76685 CBXJ07 56925623 Ki = 5600 nM T76685 C8GR5O 56925624 Ki = 5600 nM T76685 C1MIN3 56925625 Ki > 10000 nM T76685 C3N9CZ 56925626 Ki > 10000 nM T76685 C6VP7T 56925628 Ki = 1120 nM T76685 C1HO6A 56925747 Ki = 2710 nM T76685 CUB7Q2 56925748 Ki = 430 nM T76685 CHQJ12 56925749 Ki = 1860 nM T76685 C7LH9I 56925750 Ki > 10000 nM T76685 CDEM08 56925751 Ki = 3780 nM T76685 CF7QC3 56925752 Ki > 10000 nM T76685 C47TIH 56925753 Ki > 10000 nM T76685 C6X4BI 56925870 Ki = 170 nM T76685 CPS34F 56925871 Ki = 270 nM T76685 CQAD90 56925872 Ki = 2940 nM T76685 C9DS8J 56925873 Ki = 1040 nM T76685 C25PRG 56925874 Ki > 10000 nM T76685 CJ3XS5 56925875 Ki > 10000 nM T76685 COM7T4 56925978 Ki > 10000 nM T76685 C9IQJ4 56930623 Ki = 1.1 nM T76685 CG6E3T 56930624 Ki = 0.2 nM T76685 CEU17F 56930925 Ki = 25.2 nM T76685 CZ1NX6 56931060 Ki = 7.7 nM T76685 CP28UN 56931061 Ki = 66.1 nM T76685 CO6E0R 56931062 Ki = 9.4 nM T76685 CH36LK 56931063 Ki = 45.9 nM T76685 CH0ZA7 56931064 Ki = 48.7 nM T76685 CB6TF2 56931065 Ki = 3 nM T76685 CR72TI 56931190 Ki = 53.1 nM T76685 C4Q0HK 56931191 Ki = 6.7 nM T76685 C0I6QB 56931192 Ki > 10000 nM T76685 CN6J2L 56931193 Ki = 136.3 nM T76685 C9OI6H 56931194 Ki = 74.1 nM T76685 CJ86AH 56931195 Ki = 8.6 nM T76685 C08RFS 56931309 Ki = 55.6 nM T76685 CN19LG 56931310 Ki = 5.6 nM T76685 C8AGO4 56931311 Ki = 454 nM T76685 CD7T1G 56931312 Ki = 965.7 nM T76685 CR71AS 56931313 Ki = 48 nM T76685 CAM7P0 56951321 Ki = 2900 nM T76685 CW2F4U 57329634 EC50 = 913 nM T76685 C2HZB0 57341135 Ki = 39.1 nM T76685 C7C2AQ 57341136 Ki = 77.9 nM T76685 CPJ3F8 57341327 Ki = 271 nM T76685 C8S4VX 57341330 Ki = 65.5 nM T76685 C50JMF 57341331 Ki = 22.3 nM T76685 C4CI3V 57341512 Ki = 11.84 nM T76685 CJ9FN2 57341514 Ki = 97 nM T76685 C26YHM 57341678 Ki = 134 nM T76685 CIC4R1 57341679 Ki = 125 nM T76685 C6WLP1 57341681 Ki = 17.5 nM T76685 CVK8R4 57342713 Ki = 0.4 nM T76685 CGU32A 57342714 Ki = 78.4 nM T76685 CC8T6P 57342881 Ki = 42.3 nM T76685 CX1Q5W 57342882 Ki = 104 nM T76685 CX3KY7 57342883 Ki = 62.6 nM T76685 C4E5IK 57342884 Ki = 7.3 nM T76685 C6NF1A 57342885 Ki = 47.1 nM T76685 CTB1X5 57343047 Ki = 43 nM T76685 CC6T0U 57343049 Ki = 614 nM T76685 CHQU04 57343050 Ki = 1489 nM T76685 C6AS5E 57343221 Ki = 38.8 nM T76685 C5DT6K 57343222 Ki = 13.5 nM T76685 CHD82G 57343223 Ki = 15 nM T76685 C7QWP1 57343224 Ki = 7.6 nM T76685 C3QHI6 57343388 Ki = 792 nM T76685 CYE41Z 57343389 Ki = 15.5 nM T76685 CEL9T2 57343390 Ki = 2.9 nM T76685 CI5EO4 57343392 Ki = 65.3 nM T76685 C4EXK2 57343552 Ki = 14.7 nM T76685 C4TGD8 57343554 Ki = 165 nM T76685 CVR4L9 57343718 Ki = 86 nM T76685 C4JD1Z 57343719 Ki = 184 nM T76685 C80TPF 57343720 Ki = 187 nM T76685 CP5Q3T 57343721 Ki = 9.2 nM T76685 CE6RP0 57345610 Ki = 140 nM T76685 C21ZIX 57345611 Ki = 501 nM T76685 C7HU4M 57345612 Ki = 522 nM T76685 CKL7X9 57345765 IC50 = 205 nM T76685 C5K7QN 57387465 IC50 = 454 nM T76685 CEP0O6 57390497 Ki > 10000 nM T76685 CIV2U0 57390698 EC50 > 10000 nM T76685 CSV86Y 57390762 EC50 > 10000 nM T76685 CRFH16 57390958 Ki = 3 nM T76685 CNHS45 57390959 EC50 = 150 nM T76685 CG74WV 57392498 EC50 = 955 nM T76685 C4M2DZ 57392499 EC50 = 3850 nM T76685 CLD7W5 57392500 EC50 > 10000 nM T76685 C8X5TH 57393210 Ki = 60 nM T76685 CZF5C6 57394209 EC50 = 804 nM T76685 C0XDZ8 57394407 Ki = 76 nM T76685 COC84J 57394471 Ki = 22 nM T76685 CKW7S4 57396050 EC50 > 10000 nM T76685 CM5DG7 57396051 EC50 > 10000 nM T76685 C6C0IU 57396173 Ki = 592 nM T76685 CW2J4A 57396230 Ki = 264 nM T76685 CY4P3I 57396231 Ki = 32 nM T76685 C07JTI 57396232 Ki = 34 nM T76685 C80MDW 57396233 Ki = 22 nM T76685 CJT6Q5 57396515 Ki = 1.5 nM T76685 CI30KJ 57396516 Ki = 249 nM T76685 CV3I7P 57397849 EC50 = 321 nM T76685 C94JGZ 57397985 Ki = 424 nM T76685 C1TRB5 57398026 Ki = 102 nM T76685 C7HOF1 57399434 EC50 = 3630 nM T76685 CR0XE3 57399435 EC50 = 8320 nM T76685 CP6D2M 57399436 EC50 > 10000 nM T76685 C25STE 57399512 EC50 = 2676 nM T76685 C9JLX0 57399513 EC50 > 10000 nM T76685 C5UDS3 57399685 Ki = 31 nM T76685 CGA6V7 57399686 EC50 = 71 nM T76685 C5JTU0 57399687 Ki = 2380 nM T76685 CPU9O6 57401192 EC50 > 10000 nM T76685 C8SW2Q 57401265 EC50 > 10000 nM T76685 C75DTX 57401266 EC50 = 2512 nM T76685 CS4YZ9 57402953 EC50 > 10000 nM T76685 C80XAI 57403011 EC50 > 10000 nM T76685 CD2YM3 57403012 EC50 > 10000 nM T76685 CHA41T 57403138 Ki = 197 nM T76685 CO94YE 57403139 Ki = 226 nM T76685 CR52WE 57403187 EC50 = 103 nM T76685 C0BVA6 57403652 Ki = 800 nM T76685 CH24BN 57404063 EC50 = 38 nM T76685 CW48PA 57432768 Ki = 0.7943 nM T76685 CY3O0M 57441073 Ki = 11.75 nM T76685 CKOW75 57458928 Ki = 2.3 nM T76685 CP0BN7 57458937 Ki = 21 nM T76685 C41WFI 57507910 EC50 = 178 nM T76685 CIMZ13 57507911 EC50 = 54 nM T76685 CD7KI5 57555816 EC50 = 19.95 nM T76685 C7D1JL 57606048 Ki = 29.3 nM T76685 C9I6RO 57606050 EC50 = 30.7 nM T76685 CFK20V 57606063 EC50 = 1.9 nM T76685 C6D3MG 57606067 EC50 = 173 nM T76685 C3OQ4Z 57606068 EC50 = 291 nM T76685 C9V3ES 57606069 EC50 = 9.8 nM T76685 CYEQ10 57606070 EC50 = 101 nM T76685 CRDT98 57606084 Ki = 576 nM T76685 CY59ML 57606091 EC50 = 78.7 nM T76685 C1F2DJ 57606095 EC50 = 43.7 nM T76685 CIOH50 57606098 EC50 = 12.9 nM T76685 CO6F5H 57606099 Ki = 17.3 nM T76685 CLD68M 57780750 EC50 = 1.7 nM T76685 C4FNG6 57780757 EC50 = 16 nM T76685 C7LE9H 57780760 EC50 = 1.3 nM T76685 CSFA20 58124325 EC50 = 2.1 nM T76685 CT12KZ 58459056 EC50 > 100000 nM T76685 CL85HS 58459075 EC50 = 5000 nM T76685 C35EYG 58459090 EC50 > 100000 nM T76685 CV5O8N 58459093 EC50 > 100000 nM T76685 C20RBA 58459095 EC50 = 6160 nM T76685 C7AZ0L 58459098 EC50 = 1380 nM T76685 C06UDC 58459099 Ki > 1000 nM T76685 CRX0O9 58513615 EC50 > 25000 nM T76685 CO9VG5 58563756 EC50 > 20000 nM T76685 CQU7K0 58563758 EC50 = 600 nM T76685 CE4D3P 58563847 EC50 > 20000 nM T76685 CSTP80 58563862 EC50 > 20000 nM T76685 C4ZMC6 58722261 EC50 = 165 nM T76685 C2K8MN 58722274 EC50 > 10000 nM T76685 CGZ72Q 58882471 EC50 = 6 nM T76685 C50VGR 58882571 EC50 > 5000 nM T76685 CEF5R0 58973328 IC50 > 10000000 nM T76685 CV6R3G 58973346 EC50 = 180 nM T76685 CKC13R 58973398 EC50 = 5.9 nM T76685 C6ZQ3C 58973420 IC50 = 5 nM T76685 C87QCM 58973433 IC50 = 4.3 nM T76685 C1WZ9B 58999139 IC50 = 9.5 nM T76685 CDG3R9 59016064 EC50 > 3162.28 nM T76685 CH0C3G 59169713 Ki = 6.8 nM T76685 C6OSC9 59515539 Ki = 214 nM T76685 C0K2HL 59699565 Ki = 560 nM T76685 CWX31A 59718742 Ki = 1351 nM T76685 CA3X1B 59718743 Ki = 69 nM T76685 CQ90HR 59718804 Ki = 591 nM T76685 CNK4O7 59718824 Ki = 1056 nM T76685 CS4N1M 59718841 Ki = 32 nM T76685 CRFL45 59718847 Ki = 890 nM T76685 CPAJ14 59718848 Ki = 30 nM T76685 CS0W6L 59718873 Ki = 2.9 nM T76685 C6WOR7 59747725 Ki = 46.99 nM T76685 CDJ6F0 59747751 Ki = 5.998 nM T76685 CG7WN9 59799318 EC50 > 10000 nM T76685 CL5W4C 60145369 Ki = 67 nM T76685 CJ4I7K 60145370 Ki = 16.5 nM T76685 CLZ36M 60145371 Ki = 300 nM T76685 CP7H3F 60145372 Ki = 206 nM T76685 CST6V2 60145373 Ki = 1200 nM T76685 CYER47 60145524 Ki = 64.6 nM T76685 CT32WR 60145526 Ki = 234 nM T76685 C94VJI 60145527 Ki = 70 nM T76685 CAKN82 60145528 Ki > 10000 nM T76685 CK54GR 60145662 Ki = 43 nM T76685 CICU98 60145663 Ki = 950 nM T76685 C32PWF 60145664 Ki > 10000 nM T76685 CT8ED4 60145665 Ki = 1811 nM T76685 CM3C5S 60145666 Ki = 100 nM T76685 C5QS4J 60148513 Ki = 4.5 nM T76685 CE5J4O 60149000 EC50 > 100000 nM T76685 CJ6VL2 60150697 Ki = 0.08 nM T76685 C2W9BH 60150698 Ki = 0.54 nM T76685 CORL92 60154838 Ki > 10000 nM T76685 C91ITY 60154841 Ki > 10000 nM T76685 CDF8J3 60154924 Ki = 560 nM T76685 C9O4VR 60154925 Ki = 1660 nM T76685 CR8H4E 60154926 Ki = 488 nM T76685 CT3ZU0 60154927 Ki = 698 nM T76685 C0PME3 60154928 Ki = 1508 nM T76685 C1G5UC 60155009 Ki = 530 nM T76685 CP6DH5 60155010 Ki > 10000 nM T76685 CK56XU 60155011 Ki = 1827 nM T76685 C0Q7MN 60155012 Ki = 2380 nM T76685 CN8W3E 60155013 Ki > 10000 nM T76685 CRY3M4 60155101 Ki = 344.9 nM T76685 CX72BW 60155102 Ki > 10000 nM T76685 C9MGL1 60155103 Ki = 3617 nM T76685 CD5W7S 60155104 Ki = 3915 nM T76685 C5I9SG 60155105 Ki > 10000 nM T76685 C1LEX2 60155185 Ki = 48.2 nM T76685 CGBH93 60155186 Ki > 10000 nM T76685 C6TP9E 60155187 Ki = 2794 nM T76685 CBC50Z 60155188 Ki = 1052 nM T76685 CM81VH 60155189 Ki = 341.6 nM T76685 COYK60 60155275 Ki = 3621 nM T76685 CL3HG6 60155276 Ki = 2.03 nM T76685 CVA6Z1 60155280 Ki > 10000 nM T76685 CR70DY 60155369 Ki = 5510 nM T76685 C3F4XM 60155736 IC50 > 10000 nM T76685 C27XCO 60155737 IC50 > 10000 nM T76685 CEU78G 60155738 IC50 > 10000 nM T76685 CU3H4T 60155817 EC50 > 10000 nM T76685 CQ0D2Z 60155818 EC50 > 10000 nM T76685 CV6Y9Q 60155819 EC50 = 360 nM T76685 CVZ0D5 60155820 EC50 > 10000 nM T76685 C1TRU8 60155821 EC50 = 960 nM T76685 CWP04U 60155822 EC50 = 50 nM T76685 C9RH8P 60155823 EC50 = 470 nM T76685 C2LXE9 60155915 EC50 = 760 nM T76685 C0X6TB 60155916 EC50 = 4580 nM T76685 C18GHZ 60155917 IC50 > 10000 nM T76685 CHO64N 60155918 EC50 = 1510 nM T76685 C75SZK 60155919 EC50 = 230 nM T76685 CD8S3V 60155920 EC50 = 810 nM T76685 CQFG39 60155921 EC50 = 90 nM T76685 CUY1D2 60156024 EC50 > 10000 nM T76685 CACY36 60156025 IC50 > 10000 nM T76685 CF4T0W 60156026 IC50 > 10000 nM T76685 C5PFT2 60156027 EC50 = 1530 nM T76685 C6YVH8 60168041 IC50 = 120 nM T76685 C1D0WM 60168356 EC50 > 10000 nM T76685 CUP40N 60168357 EC50 > 10000 nM T76685 CZPG14 60168437 EC50 > 10000 nM T76685 CWER04 60168627 EC50 > 10000 nM T76685 CY52RD 60194851 Ki = 2866 nM T76685 C1IQ4D 60194852 Ki = 4652 nM T76685 C0J9IC 60194853 Ki > 10000 nM T76685 CNE0W5 60194854 Ki > 10000 nM T76685 CD5FM4 60194855 Ki = 105 nM T76685 CC0YJ5 60194856 Ki = 843 nM T76685 C9IPS3 60194934 Ki = 197 nM T76685 C2QP1O 60194935 Ki = 578 nM T76685 C94RWT 60194936 Ki = 88 nM T76685 C76HOR 60194937 Ki = 858 nM T76685 CPC37E 60194939 Ki > 10000 nM T76685 CKE71C 60195491 Ki = 132 nM T76685 CK4JA9 60195572 Ki = 420 nM T76685 CP0E6D 60195573 Ki = 310 nM T76685 CO0P4A 60195574 Ki = 265 nM T76685 CVX21O 60195576 Ki = 3126 nM T76685 CSL35V 60195655 Ki = 2435 nM T76685 CP1AR4 60195656 Ki > 10000 nM T76685 C4H7CW 60195657 Ki = 4108 nM T76685 CFNO62 60195658 Ki = 3877 nM T76685 CQSK90 60195659 Ki = 1346 nM T76685 CAP71F 60195741 Ki = 2150 nM T76685 CH84CF 60195742 Ki > 10000 nM T76685 C2DPQ3 60195743 Ki > 10000 nM T76685 COAS29 60195744 Ki = 821 nM T76685 C14UMZ 60195745 Ki = 433 nM T76685 C5M9SZ 60195831 Ki = 389 nM T76685 CYHG21 60195832 Ki > 10000 nM T76685 C9VD5Y 60195833 Ki = 1150 nM T76685 CWXZ73 60195835 Ki > 10000 nM T76685 C8K4BZ 60195836 Ki = 10.2 nM T76685 C74ZPK 60195919 Ki = 215 nM T76685 C3FV2S 60195921 Ki = 756 nM T76685 CV7R1C 60195922 Ki = 450 nM T76685 CSD9O4 60195923 Ki = 102 nM T76685 C5R8ZK 60195924 Ki = 91 nM T76685 CP4E9Y 60196006 Ki = 389 nM T76685 CT0JX4 60196007 Ki = 323 nM T76685 C4XG7M 60196008 Ki = 221 nM T76685 CC7XE8 60196009 Ki = 389 nM T76685 CUW84T 60196010 Ki = 1752 nM T76685 C2SU6Z 60196093 Ki = 521 nM T76685 CXZR09 60196094 Ki > 10000 nM T76685 C5BVR2 60196095 Ki > 10000 nM T76685 C2TQ6D 60196096 Ki = 105 nM T76685 CA7MG4 62705820 EC50 = 948 nM T76685 C09XDB 62705987 EC50 > 100000 nM T76685 CL92XI 62705988 EC50 > 100000 nM T76685 C8W6PJ 62705989 EC50 > 100000 nM T76685 CUE8H3 64428131 Ki = 2700 nM T76685 CKV0W6 66546152 IC50 = 3 nM T76685 CQ40JT 66546337 IC50 = 15 nM T76685 CKRE08 66546338 IC50 = 22 nM T76685 C7X6KT 66546339 IC50 = 21 nM T76685 C0VWQ5 66546340 IC50 > 1000 nM T76685 CDQS32 66546341 IC50 = 33 nM T76685 CLAD79 66546526 IC50 = 4 nM T76685 COJ0M9 66546527 IC50 = 12 nM T76685 CIL1S2 66546529 IC50 = 137 nM T76685 CTV3B0 66546530 IC50 > 1000 nM T76685 CMX68Q 66546531 IC50 = 9 nM T76685 C7I1HB 66546710 IC50 = 112 nM T76685 CC97QD 66546711 IC50 = 10 nM T76685 COKD45 66546713 IC50 = 12 nM T76685 CJ79QL 66546714 IC50 = 10 nM T76685 C8V3KQ 66546715 IC50 = 4 nM T76685 CT8MI9 66546894 IC50 = 15 nM T76685 CDQ46S 66546895 IC50 = 3 nM T76685 C9HR4P 66546896 IC50 = 3 nM T76685 CN2V3I 66546897 IC50 = 41 nM T76685 CF30UC 66546899 IC50 = 7 nM T76685 CV8G6N 66546900 IC50 = 5 nM T76685 C40BQL 66547072 IC50 = 2 nM T76685 C3W5GS 66547074 IC50 = 6 nM T76685 C4DSE6 66547075 IC50 = 2 nM T76685 CPE3F6 66547076 IC50 = 200 nM T76685 C9ZE0C 66547078 IC50 > 1000 nM T76685 CFT7Z0 66547239 IC50 = 500 nM T76685 CL94XN 66547240 IC50 = 130 nM T76685 C4A2PD 66547241 IC50 > 200 nM T76685 C6OXE5 66547242 IC50 > 1000 nM T76685 C69UHC 66547243 IC50 = 800 nM T76685 C3VTQ1 66547244 IC50 = 800 nM T76685 CI1YE4 66547245 IC50 > 1000 nM T76685 C10FRE 66547410 IC50 = 8 nM T76685 CF9W1L 66547411 IC50 > 1000 nM T76685 C7CFE5 66547412 IC50 = 200 nM T76685 CV5Q7E 66547413 IC50 = 400 nM T76685 C6WSU0 66547414 IC50 = 250 nM T76685 CW5Q0G 66547415 IC50 = 200 nM T76685 C08LFD 66547416 IC50 = 500 nM T76685 C96IAU 66547417 IC50 > 1000 nM T76685 C7JLO5 66547588 IC50 = 300 nM T76685 C9XL5J 66547589 IC50 = 200 nM T76685 CR8V2Y 66553217 IC50 = 2 nM T76685 CUA9G5 66643149 EC50 > 27000 nM T76685 CTS7P8 67012376 Ki = 23.5 nM T76685 CKZO03 67425523 EC50 > 100000 nM T76685 C8YE5J 67425691 EC50 > 100000 nM T76685 CVZP79 67427023 EC50 > 1000000 nM T76685 CLS9K6 67433936 EC50 = 1430 nM T76685 C9YZR3 67434101 EC50 = 6160 nM T76685 C0LGO7 67434539 EC50 = 512 nM T76685 C09VFU 67434704 EC50 > 100000 nM T76685 CL8QT1 67435171 EC50 = 4770 nM T76685 CML5F8 67450266 EC50 = 13300 nM T76685 C8Q9MN 67455563 EC50 = 54 nM T76685 CT1E8P 67457326 EC50 > 20000 nM T76685 CD40IL 67458256 EC50 > 20000 nM T76685 CXQ85N 67505405 Ki = 1074 nM T76685 C6W1UQ 67519772 Ki = 266 nM T76685 C9KZ7X 67520157 Ki = 1877 nM T76685 CX1AL0 67520222 IC50 = 76 nM T76685 C4H6ZJ 67520284 Ki > 5000 nM T76685 CX3Z9O 67953246 EC50 > 50000 nM T76685 CPB54A 67953263 EC50 = 28000 nM T76685 CI13QS 67953265 EC50 > 50000 nM T76685 CZP98A 67953277 EC50 = 29000 nM T76685 CE94JQ 67953283 EC50 = 30 nM T76685 C3T6JM 67953286 EC50 > 20000 nM T76685 C06ADK 67953287 EC50 = 15 nM T76685 CR9BV5 67953290 EC50 > 20000 nM T76685 CBK74Z 67953291 EC50 > 20000 nM T76685 C19YPW 67953294 EC50 = 41000 nM T76685 C2D6XA 67953297 EC50 = 4900 nM T76685 CX3E4U 67953298 EC50 = 7200 nM T76685 C42TIW 67953300 EC50 = 10100 nM T76685 C5JUY1 67953301 EC50 = 98005 nM T76685 CXI91V 67953302 EC50 = 2400 nM T76685 CMYD72 67953303 EC50 = 390 nM T76685 C0I5FH 67953329 EC50 > 50000 nM T76685 CT43SM 67953330 EC50 > 50000 nM T76685 CUB95N 67953333 EC50 > 50000 nM T76685 CH7FG3 67953351 EC50 > 50000 nM T76685 C3YQN6 67953380 EC50 > 20000 nM T76685 C0DP2O 67953418 EC50 = 970 nM T76685 C0T2AG 67953425 EC50 = 3200 nM T76685 CX01CP 67953431 EC50 = 110 nM T76685 CX13CH 67953836 EC50 = 7 nM T76685 CPTA39 67953837 EC50 = 307 nM T76685 C4XKL9 67953838 EC50 > 20000 nM T76685 CIHR82 67953851 EC50 = 53 nM T76685 CGC79J 67953920 EC50 = 1100 nM T76685 CI86RD 67956378 Ki = 176 nM T76685 C3S6AU 67970610 Ki = 104 nM T76685 CL4K0D 68160786 Ki = 548 nM T76685 CSIR78 68182311 EC50 > 30000 nM T76685 C7CSY1 68182368 EC50 > 30000 nM T76685 CPG5Q9 68278877 Ki > 10000 nM T76685 C30INO 68353389 EC50 > 10000 nM T76685 C6BG0N 68555650 EC50 > 27000 nM T76685 C8PN7J 68603000 EC50 = 22900 nM T76685 C9Q1KW 68603392 EC50 = 6050 nM T76685 CCQ6V1 68603806 EC50 > 100000 nM T76685 C8BS2C 68604012 EC50 > 100000 nM T76685 CN2T0C 68604144 EC50 > 100000 nM T76685 CJ94SD 68604381 EC50 = 16900 nM T76685 CGE5X2 68604800 EC50 > 100000 nM T76685 C45DZE 68604816 EC50 = 3010 nM T76685 CAN1O3 68741582 Ki = 8880 nM T76685 C46DPY 68742556 Ki = 480 nM T76685 CZL35B 68904230 Ki > 10000 nM T76685 C5GLN7 68908342 Ki > 10000 nM T76685 C75UTD 68908346 Ki = 1905.46 nM T76685 C84XYG 68909935 Ki > 10000 nM T76685 CJVP65 68910242 Ki > 10000 nM T76685 C1XPM0 69003787 IC50 = 3881 nM T76685 CIZD23 69007013 EC50 > 17000 nM T76685 C0WAL2 69111813 Ki = 4585 nM T76685 CNQH46 69240356 IC50 = 95 nM T76685 C1CY2U 69307211 Ki = 29 nM T76685 C3XV4P 69472197 Ki > 5000 nM T76685 C1L3WU 69474974 Ki = 3952 nM T76685 C84XJE 69475608 Ki > 5000 nM T76685 CC9IR4 69488978 EC50 = 199.53 nM T76685 C59YDO 69489075 EC50 = 158.49 nM T76685 C4NM1C 69493574 Ki = 6.3 nM T76685 CLG7R1 69516364 EC50 = 316.23 nM T76685 C2AZ4X 69787126 IC50 = 63.1 nM T76685 C0YH3T 70677671 Ki > 10000 nM T76685 CQT54O 70677672 Ki = 21100 nM T76685 CR71AY 70677673 Ki > 10000 nM T76685 C8VQ0M 70677674 Ki = 4740 nM T76685 CURQ38 70677675 Ki > 10000 nM T76685 CGR4U7 70677676 Ki > 10000 nM T76685 CFMD45 70677677 Ki = 45 nM T76685 C2E1AD 70677804 Ki = 16200 nM T76685 CVX9I7 70677805 Ki = 1920 nM T76685 CLWV92 70677806 Ki = 1270 nM T76685 CCE2U9 70677807 Ki = 22 nM T76685 C74KDW 70677808 Ki = 1640 nM T76685 CK4C2I 70677809 Ki = 713 nM T76685 CTYE29 70677810 Ki = 2170 nM T76685 CSGH58 70677953 Ki = 32 nM T76685 CY3O0R 70677954 Ki = 9820 nM T76685 CCUW05 70677955 Ki = 33 nM T76685 CB4P6Y 70677956 Ki = 19100 nM T76685 C6ESV8 70677957 Ki = 637 nM T76685 C3F2AY 70677958 Ki = 6390 nM T76685 CV7Q3G 70677959 Ki = 1430 nM T76685 C4Y1LE 70678097 Ki = 2630 nM T76685 C3DX1U 70678098 Ki = 1020 nM T76685 C71DQG 70678099 Ki = 244 nM T76685 CJ0P4V 70678100 Ki = 10000 nM T76685 C82PMZ 70678101 Ki = 1170 nM T76685 CTB19O 70678102 Ki = 598 nM T76685 C46QGZ 70678238 Ki = 1580 nM T76685 CBX9D4 70678239 Ki >= 10000 nM T76685 CS7FL4 70678240 Ki = 4890 nM T76685 C30LIP 70678241 Ki > 10000 nM T76685 CT1EF6 70678242 Ki > 10000 nM T76685 CT9C3E 70681203 EC50 = 31.62 nM T76685 CP0H4S 70681204 EC50 = 630.96 nM T76685 CO7SP4 70681279 Ki = 39 nM T76685 CZ3X4M 70681392 IC50 = 297 nM T76685 C0SVD9 70681412 IC50 > 2000 nM T76685 CO78DU 70683293 EC50 = 1258.93 nM T76685 C63YFK 70683294 EC50 = 1000 nM T76685 C2MSC9 70683383 Ki > 5000 nM T76685 C8LN6Z 70683449 Ki = 109 nM T76685 C4YUC3 70684359 Ki = 0.56 nM T76685 C3IXK2 70684360 Ki = 0.26 nM T76685 CK6NA5 70685024 IC50 > 10000 nM T76685 C4IRK6 70685401 EC50 = 79.43 nM T76685 CTD3I6 70685551 Ki = 4.6 nM T76685 C65WEJ 70686524 Ki = 0.03 nM T76685 C1UFM2 70687544 EC50 = 158.49 nM T76685 CA4UM9 70687741 IC50 = 657 nM T76685 C8WKV5 70687770 IC50 = 291 nM T76685 CJ0Z2Y 70687771 IC50 = 398 nM T76685 CJ6KE0 70687772 IC50 = 23 nM T76685 C13TJG 70689601 EC50 = 158.49 nM T76685 C8GR7P 70689602 EC50 = 2511.89 nM T76685 CJMG21 70689659 Ki = 3.4 nM T76685 C2BA8P 70689660 Ki = 8 nM T76685 CSI98P 70689667 Ki = 218 nM T76685 C6UVC8 70689694 IC50 = 468 nM T76685 C3L1HS 70689695 IC50 = 113 nM T76685 CN43EU 70689696 IC50 > 2000 nM T76685 CQ95RM 70689788 IC50 = 611 nM T76685 CXO85R 70689820 IC50 > 2000 nM T76685 C7UJ0Y 70690691 Ki = 5.1 nM T76685 CGOP85 70690692 Ki = 0.07 nM T76685 C6K9DE 70690693 Ki = 1.4 nM T76685 CF0TP8 70691731 EC50 = 630.96 nM T76685 CQYA93 70691732 EC50 = 501.19 nM T76685 C8OLN3 70691798 Ki = 5.8 nM T76685 C5XZR6 70691799 Ki = 242 nM T76685 CYO5G4 70692838 Ki = 0.23 nM T76685 CKDW02 70692839 Ki = 4.3 nM T76685 CS63PK 70693593 Ki > 10000 nM T76685 CL06EQ 70693862 Ki = 4.7 nM T76685 CT7Q5W 70693863 Ki = 11 nM T76685 CW8LU2 70693864 Ki = 4.9 nM T76685 C4T9MB 70693933 Ki = 52 nM T76685 CY4CH9 70694009 IC50 = 997 nM T76685 CX2NM7 70694867 Ki = 0.05 nM T76685 CE7W2O 70694868 Ki = 0.08 nM T76685 C1PDK2 70695982 Ki = 2970 nM T76685 C6YG8R 70696000 IC50 > 2000 nM T76685 C1FU9R 70696001 Ki > 5000 nM T76685 C8R3JH 70696105 Ki = 34 nM T76685 CL6WD5 70696134 IC50 > 2000 nM T76685 CB50NG 70696261 EC50 = 70.6 nM T76685 CUS64H 70864970 EC50 > 20000 nM T76685 CN5G3Z 70864972 EC50 = 6979 nM T76685 CA8CQ4 70865076 EC50 = 15640 nM T76685 C2PJ1D 70865101 EC50 > 20000 nM T76685 C5H8UT 70865109 EC50 > 20000 nM T76685 CUY4E2 70865116 EC50 > 20000 nM T76685 CQX01V 70865117 EC50 = 7895 nM T76685 CR13JM 70865325 EC50 > 20000 nM T76685 C4OK5W 70865326 EC50 > 20000 nM T76685 C90OTR 70865329 EC50 > 20000 nM T76685 CBTY34 71020062 Ki > 10000 nM T76685 C1NYW6 71116224 Ki = 6.4 nM T76685 CU5NM8 71138232 EC50 > 100000 nM T76685 CR12DH 71138284 EC50 = 4660 nM T76685 CEK26Z 71138285 EC50 = 4660 nM T76685 C7EZS4 71301472 EC50 = 2.1 nM T76685 CVQ1T2 71308155 EC50 = 39 nM T76685 C83XZQ 71308243 Ki = 245 nM T76685 CY8KL0 71449129 IC50 = 2.8 nM T76685 CCH78A 71449130 IC50 = 3.4 nM T76685 CEMC56 71449131 IC50 = 14 nM T76685 CD35HU 71449370 Ki > 3000 nM T76685 CPL4J3 71449371 Ki > 1000 nM T76685 C9NHQ5 71449464 Ki = 193 nM T76685 CAY6E5 71449465 Ki = 4 nM T76685 CF0HK8 71449466 Ki = 28.8 nM T76685 CCYF04 71449467 Ki = 20.9 nM T76685 CDT13U 71449468 Ki = 58.2 nM T76685 CSOD75 71449527 IC50 > 5000 nM T76685 CHW0A3 71449530 IC50 = 8.3 nM T76685 CAYC78 71449541 IC50 = 13 nM T76685 C0MN4L 71449542 IC50 = 4 nM T76685 C8P3SF 71449726 Ki = 200 nM T76685 CWDN02 71450141 Ki > 20000 nM T76685 C98YPR 71450142 Ki = 109 nM T76685 CN5SC9 71450187 Ki = 14 nM T76685 C2S6LQ 71450188 Ki = 11 nM T76685 C0ZT2Y 71450189 Ki = 25.5 nM T76685 CT83NB 71450463 EC50 = 217 nM T76685 C8W2GK 71450464 EC50 = 81 nM T76685 CLDY61 71450465 EC50 = 113 nM T76685 C0DG7B 71450466 EC50 = 3217 nM T76685 C1EN0J 71450467 EC50 > 10000 nM T76685 CYT1Z2 71450516 EC50 = 9360 nM T76685 C9S8IF 71450517 EC50 > 10000 nM T76685 C2GOT7 71450518 EC50 = 6611 nM T76685 CI1L7R 71450519 EC50 = 1905 nM T76685 CN96YC 71450520 EC50 > 10000 nM T76685 C35AKH 71450521 EC50 > 10000 nM T76685 C1BJ9N 71450522 EC50 > 10000 nM T76685 C9FY0A 71450641 Ki = 2960 nM T76685 CZJV01 71450642 Ki = 187 nM T76685 CV90CJ 71450643 Ki = 8.9 nM T76685 C85ANU 71451170 Ki > 3000 nM T76685 C60ILF 71451171 Ki > 3000 nM T76685 C75VXY 71451172 Ki > 3000 nM T76685 CAWS56 71451265 Ki = 178.7 nM T76685 CYU28K 71451266 Ki = 3572.6 nM T76685 C90EMT 71451267 Ki = 4.7 nM T76685 CH1QU4 71451268 Ki > 10000 nM T76685 C7YM3V 71451269 Ki = 28.9 nM T76685 C2D3EN 71451270 Ki = 63.2 nM T76685 CYD6H5 71451324 IC50 = 20 nM T76685 CI1DG5 71451325 IC50 > 100 nM T76685 C1EL7T 71451331 IC50 = 66 nM T76685 C8J1YK 71451332 IC50 > 500 nM T76685 CDJO69 71451333 IC50 = 27 nM T76685 C7NS9H 71451521 Ki > 10000 nM T76685 CDES68 71451522 Ki > 10000 nM T76685 CB9MI7 71451970 Ki > 20000 nM T76685 CHN2J6 71451971 Ki > 20000 nM T76685 C6XJ3A 71451973 Ki > 20000 nM T76685 C9WSP6 71451974 Ki > 20000 nM T76685 C65FUD 71451975 Ki > 20000 nM T76685 CE5H8L 71451976 Ki > 20000 nM T76685 CVUQ43 71452011 Ki = 25 nM T76685 C4POZ7 71452013 Ki = 269 nM T76685 CM8X9C 71452295 EC50 = 958 nM T76685 CROF14 71452296 EC50 > 10000 nM T76685 CLW23T 71452368 EC50 = 243 nM T76685 CFH25Z 71452369 EC50 > 10000 nM T76685 CA8MB6 71452370 EC50 = 251 nM T76685 CM17YT 71452371 EC50 = 812 nM T76685 C01EHK 71452372 EC50 = 4639 nM T76685 C3WB7F 71452473 Ki = 14 nM T76685 CZ65ND 71452474 Ki = 642 nM T76685 CU0C6V 71452475 Ki = 161 nM T76685 C3M6NR 71452739 IC50 = 12 nM T76685 CO73CM 71452740 IC50 = 33 nM T76685 CA0IP1 71453003 Ki > 3000 nM T76685 CF53WM 71453004 Ki > 1000 nM T76685 C96RTE 71453082 Ki = 296.8 nM T76685 C9SN8B 71453083 Ki = 398.5 nM T76685 CUW47P 71453084 Ki = 11 nM T76685 C1S4AY 71453085 Ki = 390 nM T76685 COV6P0 71453086 Ki = 86.6 nM T76685 CT2AJ3 71453087 Ki = 1490 nM T76685 CI13LY 71453088 Ki = 490 nM T76685 C3ND5C 71453142 IC50 > 100 nM T76685 C5B4UC 71453148 IC50 = 70 nM T76685 CJ4LV0 71453149 IC50 > 100 nM T76685 C2R8FM 71453477 Ki > 1000 nM T76685 CL1R2P 71453777 Ki > 20000 nM T76685 C58LXU 71453778 Ki > 20000 nM T76685 CP86RY 71453779 Ki > 20000 nM T76685 CMWD96 71453780 Ki > 20000 nM T76685 CC73DS 71453820 Ki = 1.79 nM T76685 C59BKG 71454089 EC50 > 10000 nM T76685 CRZ5O1 71454090 EC50 = 3972 nM T76685 CEFK54 71454091 EC50 > 10000 nM T76685 CC15FR 71454137 EC50 > 10000 nM T76685 CI87XN 71454138 EC50 > 10000 nM T76685 CC7HZ4 71454139 EC50 = 5960 nM T76685 CO2D9I 71454140 EC50 = 80 nM T76685 CZE87R 71454141 EC50 = 7452 nM T76685 C25MZX 71454142 EC50 > 10000 nM T76685 CK1L0A 71454143 EC50 > 10000 nM T76685 C7RI0X 71454144 EC50 > 10000 nM T76685 C5TDX4 71454145 EC50 = 1000 nM T76685 CXY23Z 71454233 Ki = 1.2 nM T76685 C87ZBR 71454234 Ki = 73 nM T76685 CJGD87 71454235 Ki = 530 nM T76685 C6Z9KB 71454236 Ki = 7.2 nM T76685 C35CMH 71454823 Ki > 10000 nM T76685 CK5Z8D 71454824 Ki = 38.6 nM T76685 C2CFA3 71454877 IC50 = 100 nM T76685 C1OC6X 71454884 IC50 = 10 nM T76685 CX36YH 71454885 IC50 = 7 nM T76685 C2JYF6 71455057 Ki = 3120 nM T76685 C81WIN 71455077 Ki = 460 nM T76685 CJ4DG1 71455514 Ki > 20000 nM T76685 C0HA7N 71455515 Ki > 20000 nM T76685 CCR74A 71455516 Ki > 20000 nM T76685 C9OT7E 71455518 Ki > 20000 nM T76685 C1LS5H 71455552 Ki = 7.1 nM T76685 C2XH7I 71455827 EC50 = 336 nM T76685 CFJK21 71455875 EC50 = 1974 nM T76685 CSHB15 71455876 EC50 = 1500 nM T76685 CEJ2T3 71455989 Ki > 10000 nM T76685 CX54OE 71456254 IC50 = 90 nM T76685 C68CNX 71456598 Ki = 23.8 nM T76685 CKTP96 71456599 Ki > 10000 nM T76685 C7HW1G 71456600 Ki = 660 nM T76685 C0QSJ4 71456601 Ki = 12.9 nM T76685 C0NV6W 71456602 Ki > 10000 nM T76685 CD21BS 71456648 IC50 > 5000 nM T76685 C71XMI 71456649 IC50 > 5000 nM T76685 C9LOZ3 71456650 IC50 = 7 nM T76685 CNS3L4 71456661 IC50 = 8 nM T76685 C1D6KG 71456857 Ki > 10000 nM T76685 CP1OY9 71456858 Ki > 10000 nM T76685 CP4K8E 71456859 Ki = 550 nM T76685 C53VGN 71457303 Ki > 20000 nM T76685 CFG6E0 71457306 Ki > 20000 nM T76685 CW79ZE 71457341 Ki = 28 nM T76685 CKWG06 71457342 Ki = 195 nM T76685 CHF86C 71457343 Ki = 24 nM T76685 C6AWM3 71457619 EC50 > 10000 nM T76685 CID47K 71457677 EC50 = 16 nM T76685 C6LYF4 71457678 EC50 = 798 nM T76685 COS48L 71457679 EC50 = 125 nM T76685 C5G7LZ 71457680 EC50 = 8710 nM T76685 CQH74V 71457790 Ki = 373 nM T76685 CS3XD2 71457791 Ki = 2.5 nM T76685 CT90JC 71457792 Ki = 54 nM T76685 CGO45N 71457793 Ki = 4290 nM T76685 C0JP3H 71457794 Ki = 14 nM T76685 C8FGC1 71458061 IC50 = 140 nM T76685 CJ6N5E 71458352 Ki > 3000 nM T76685 CL1KS5 71458353 Ki > 3000 nM T76685 CU4RF3 71458354 Ki > 3000 nM T76685 CM2N8G 71458457 Ki = 669.3 nM T76685 CBY8N2 71458500 IC50 > 5000 nM T76685 CZA80U 71458501 IC50 > 5000 nM T76685 CG78IJ 71458502 IC50 > 1000 nM T76685 C3NJ7W 71458503 IC50 > 1000 nM T76685 C6S4RO 71458508 IC50 > 100 nM T76685 CH7L4U 71458714 Ki > 10000 nM T76685 C35XHD 71458715 Ki = 2570 nM T76685 C9SUN1 71459136 Ki > 20000 nM T76685 CUP6O2 71459139 Ki > 20000 nM T76685 C4O9AG 71459140 Ki > 20000 nM T76685 CEK2A3 71459141 Ki > 20000 nM T76685 CU1YC4 71459143 Ki > 20000 nM T76685 CKME06 71459192 Ki = 1.5 nM T76685 CGF62Y 71459194 Ki = 6.2 nM T76685 C51CZF 71459196 Ki = 3343 nM T76685 CT2YD6 71459512 EC50 = 139 nM T76685 CA46PX 71459513 EC50 > 10000 nM T76685 CY1HJ8 71459578 EC50 > 10000 nM T76685 CSA07B 71459579 EC50 = 1416 nM T76685 CI4W2B 71459580 EC50 = 296 nM T76685 CNG46Q 71459581 EC50 > 10000 nM T76685 CM8U2X 71459582 EC50 = 4538 nM T76685 C4Q3VE 71459583 EC50 = 3270 nM T76685 CIS71D 71459709 Ki = 240 nM T76685 CUQK68 71459945 IC50 = 16.98 nM T76685 C97TBJ 71460194 Ki > 3000 nM T76685 C1K6MS 71460195 Ki > 3000 nM T76685 CU3W9O 71460308 Ki = 959.7 nM T76685 C0GF4X 71460309 Ki = 14.4 nM T76685 CZT47C 71460310 Ki = 1866.9 nM T76685 C4FD5O 71460311 Ki = 2.45 nM T76685 C84SOK 71460312 Ki = 151.1 nM T76685 C4T8BN 71460313 Ki = 420 nM T76685 C6IA5P 71460345 IC50 > 1000 nM T76685 CDLM90 71460346 IC50 > 1000 nM T76685 CV6C0O 71460352 IC50 > 100 nM T76685 C1M8KG 71460548 Ki = 1365 nM T76685 C8TE6M 71460655 Ki = 87.9 nM T76685 CNA5B4 71460951 Ki > 20000 nM T76685 CC64PU 71460953 Ki > 20000 nM T76685 CWZ13R 71460978 Ki = 1.2 nM T76685 C82PAR 71460979 Ki = 337 nM T76685 C25NCA 71461256 EC50 > 10000 nM T76685 CZ94DS 71461257 EC50 > 10000 nM T76685 COT0U9 71461320 EC50 = 368 nM T76685 CS8Y2Z 71461321 EC50 = 1656 nM T76685 C02PKW 71461322 EC50 > 10000 nM T76685 CO7MH0 71461323 EC50 > 10000 nM T76685 C40DFP 71461324 EC50 > 10000 nM T76685 CP6YI3 71461325 EC50 = 1753 nM T76685 CCV94E 71461421 Ki > 10000 nM T76685 C09VOG 71461422 Ki = 93 nM T76685 CEM06G 71461910 Ki > 3000 nM T76685 CF9AQ4 71462003 Ki > 10000 nM T76685 CV9M1I 71462004 Ki = 181.3 nM T76685 C08TZO 71462005 Ki > 10000 nM T76685 CGL5O1 71462046 IC50 = 300 nM T76685 CK7FA6 71462047 IC50 = 2 nM T76685 CVB2R9 71462053 IC50 > 100 nM T76685 C1VOK3 71462054 IC50 = 100 nM T76685 CBM3S6 71462240 Ki > 10000 nM T76685 CG16QI 71462668 Ki > 20000 nM T76685 CX25GM 71462669 Ki > 20000 nM T76685 CM27NV 71462714 Ki = 29 nM T76685 CRNO72 71462715 Ki = 220 nM T76685 CE7O6K 71462979 EC50 > 10000 nM T76685 CG25YZ 71463044 EC50 = 8030 nM T76685 C3RK6B 71463045 EC50 > 10000 nM T76685 C0U5IW 71463046 EC50 > 10000 nM T76685 CU2W0X 71463047 EC50 = 607 nM T76685 CE0BD5 71463048 EC50 = 925 nM T76685 CER92U 71463049 EC50 = 519 nM T76685 C6RIO7 71463050 EC50 > 10000 nM T76685 CEO29S 71463152 Ki = 14 nM T76685 CG9HX2 71463153 Ki > 10000 nM T76685 C1QTI4 71463154 Ki = 23 nM T76685 CH3W2U 71463155 Ki = 116 nM T76685 CP26EI 71539529 Ki = 61 nM T76685 C94GWF 71539530 Ki = 275 nM T76685 C8MFO7 71539582 Ki > 60000 nM T76685 CC7QJ5 71539583 Ki = 3200 nM T76685 CIY1E4 71539585 EC50 > 30000 nM T76685 CK7OC8 71539693 Ki > 60000 nM T76685 C1I8AV 71539696 Ki > 60000 nM T76685 CHM1K5 71539697 Ki > 60000 nM T76685 CKGT70 71539698 Ki > 10000 nM T76685 C7XLD6 71539749 Ki > 10000 nM T76685 C4UN2K 71539750 Ki > 60000 nM T76685 C32GUW 71544705 EC50 = 5.9 nM T76685 C9N7YA 71544706 EC50 = 13 nM T76685 C92NEY 71544707 IC50 = 49 nM T76685 C7EMT1 71544708 IC50 = 21 nM T76685 C9P2DB 71544873 IC50 = 600 nM T76685 C0L9ON 71545855 EC50 = 260 nM T76685 C4N3OC 71545856 EC50 = 5.1 nM T76685 CV5E9K 71546015 IC50 > 10000 nM T76685 CJ75FS 71546180 IC50 = 1200 nM T76685 C6W5VM 71546181 IC50 > 9900 nM T76685 C5JD2B 71546182 IC50 = 320 nM T76685 CQJE12 71546834 EC50 = 120 nM T76685 C29NBP 71546835 EC50 = 14 nM T76685 C1IR3O 71559417 EC50 > 10000 nM T76685 C1R6XV 71559418 EC50 > 10000 nM T76685 CM56QN 71559419 EC50 > 10000 nM T76685 C7LK1F 71559522 EC50 > 10000 nM T76685 CZYK61 71559523 EC50 > 10000 nM T76685 CQ20NX 71559524 EC50 > 10000 nM T76685 CP5HX4 71559525 EC50 > 10000 nM T76685 C5DRB3 71559526 EC50 > 10000 nM T76685 CMT2O6 71559637 EC50 > 10000 nM T76685 C40KSJ 71559638 EC50 > 10000 nM T76685 CEXC24 71559639 EC50 > 10000 nM T76685 C10SJV 71559641 EC50 > 10000 nM T76685 CK57LU 71561577 Ki = 523 nM T76685 C2ZT8O 71562536 Ki = 500 nM T76685 CV6D0B 71562537 Ki = 1256 nM T76685 CDOC40 71562538 Ki = 758 nM T76685 C5VMJ8 71562539 Ki > 10000 nM T76685 C9O0IY 71562646 Ki > 10000 nM T76685 CR5DA3 71562647 Ki > 10000 nM T76685 C8Q3TG 71562648 Ki = 3870 nM T76685 CJH90S 71562649 Ki = 4248 nM T76685 CW8UR7 71562650 Ki > 10000 nM T76685 CDL5T4 71562651 Ki > 10000 nM T76685 CVW4E9 71562652 Ki = 1124 nM T76685 CFU7J4 71562780 Ki = 723 nM T76685 CFC4X3 71562781 Ki = 252 nM T76685 C8XO4U 71562782 Ki = 800 nM T76685 CBQ4R3 71562784 Ki = 1795 nM T76685 C8WGI2 71562897 Ki = 865 nM T76685 CCZ60L 71562898 Ki > 10000 nM T76685 CD37US 71562899 Ki > 10000 nM T76685 CV8Y9G 71562900 Ki > 10000 nM T76685 CUIY12 71562901 Ki = 957 nM T76685 CIX50M 71562902 Ki = 440 nM T76685 CF0HO4 71563025 Ki > 10000 nM T76685 C6PKB2 71563026 Ki = 3753 nM T76685 CNG41L 71563027 Ki = 5150 nM T76685 CR9X5F 71563028 Ki = 4550 nM T76685 CJE6L8 71563029 Ki = 4752 nM T76685 CBN0L8 71563030 Ki > 10000 nM T76685 C6T1CA 71563145 Ki > 10000 nM T76685 CMGT96 71563146 Ki > 10000 nM T76685 CE7M3O 71563147 Ki > 10000 nM T76685 C6TK3A 71563148 Ki = 155 nM T76685 CM48BC 71563149 Ki = 145 nM T76685 CY6IM3 71563150 Ki = 1468 nM T76685 CG4K6V 71563277 Ki = 86 nM T76685 CC31QD 71563278 Ki = 52 nM T76685 CZ7FL2 71563279 Ki = 13.7 nM T76685 C9M8XO 71563280 Ki = 43 nM T76685 C98DXW 71563282 Ki = 712 nM T76685 CJK19B 71580293 IC50 = 300 nM T76685 CS21CO 71583291 Ki = 6157 nM T76685 CX0JF3 71583401 Ki > 40000 nM T76685 CS52BT 71583402 Ki > 40000 nM T76685 CNAX48 71583403 Ki > 40000 nM T76685 C3LND0 71583404 Ki > 40000 nM T76685 CM09HD 71583405 Ki > 40000 nM T76685 C7BTX6 71583521 Ki > 10000 nM T76685 C78ZRD 71583522 Ki = 9690 nM T76685 C94AJQ 71583523 Ki > 40000 nM T76685 C30RXC 71583524 Ki > 10000 nM T76685 C9C2YD 71583608 Ki = 11000 nM T76685 CPC06E 71583609 Ki = 4268 nM T76685 CQBV09 71583610 Ki = 2033 nM T76685 C35QNI 71583711 Ki = 7300 nM T76685 C7DET3 71583712 Ki > 20000 nM T76685 CLTK19 71583713 Ki = 8224 nM T76685 C30KRJ 71583715 Ki > 20000 nM T76685 C1K7LR 71583828 Ki > 20000 nM T76685 CM9N3D 71583829 Ki > 20000 nM T76685 CNWE02 71584050 Ki = 1773 nM T76685 CKB0G2 71584155 Ki = 1126 nM T76685 CED16K 71584156 Ki = 6617 nM T76685 CD9QX6 71584157 Ki > 20000 nM T76685 CJQY30 71584158 Ki = 137 nM T76685 CJ58HL 71584159 Ki = 866 nM T76685 C4TL1Z 71584275 Ki > 2000 nM T76685 CLZX28 71584276 Ki > 20000 nM T76685 CE7A4L 71584277 Ki = 514 nM T76685 C3ILW7 71584278 Ki = 858 nM T76685 CF4RV8 71584279 Ki = 412 nM T76685 C2W1IH 71584410 Ki = 437 nM T76685 CZH52F 71584411 Ki = 218 nM T76685 CI0E4G 71584412 Ki = 3365 nM T76685 C6C8TB 71584413 Ki > 20000 nM T76685 CV26EB 71584414 Ki = 3200 nM T76685 C0T9US 71584415 Ki = 202 nM T76685 CMYO23 71587360 Ki = 5 nM T76685 C5YQ2V 71599710 IC50 = 180 nM T76685 C8VCB9 71623045 EC50 > 10000 nM T76685 C3UG6H 71623046 EC50 = 260 nM T76685 C3F6ES 71623048 EC50 = 1600 nM T76685 C0Z5QS 71623175 Ki = 1300 nM T76685 C5AX6I 71623227 Ki = 520 nM T76685 C7W6YB 71623228 Ki = 690 nM T76685 CG9X8V 71623343 Ki = 430 nM T76685 C03LQH 71623344 Ki = 930 nM T76685 CN7VC0 71624052 Ki = 2300 nM T76685 CBS46L 71624056 Ki = 2250 nM T76685 C1G8AO 71624057 Ki = 560 nM T76685 CS3J0O 71624058 Ki = 570 nM T76685 CAMI85 71624059 Ki = 610 nM T76685 CRY61V 71624060 Ki = 81 nM T76685 CXS93U 71624177 Ki = 340 nM T76685 C46VIA 71624178 Ki = 500 nM T76685 CAQ3Z2 71624179 Ki = 1250 nM T76685 CZR79M 71624180 Ki = 500 nM T76685 C83JIM 71624181 Ki = 2000 nM T76685 CUD56P 71624182 Ki = 840 nM T76685 C80NJP 71624301 Ki = 210 nM T76685 C85TFY 71624302 Ki = 1300 nM T76685 CU1I6J 71624303 Ki = 660 nM T76685 CO3LE7 71624304 Ki = 1400 nM T76685 C3O7BW 71624305 Ki = 600 nM T76685 CJ57PR 71624543 Ki = 590 nM T76685 CAY05V 71660059 Ki = 606 nM T76685 CSI3T7 71660060 Ki = 143 nM T76685 C3ESZ4 71660061 Ki = 746 nM T76685 CVGZ69 71660103 Ki = 9 nM T76685 CXFA37 71660104 Ki = 1769 nM T76685 CI0GU8 71660496 IC50 > 48500 nM T76685 CB9FL3 71661716 EC50 = 1.29 nM T76685 CH0E7F 71662074 EC50 = 230 nM T76685 C65QMB 71662076 EC50 = 7.97 nM T76685 C7N2BM 71680717 Ki = 120 nM T76685 CJK5C9 71680718 Ki = 675 nM T76685 CB7N4D 71680719 Ki = 605 nM T76685 CZ2OI1 71680720 Ki = 612 nM T76685 CTHM04 71680721 Ki = 702 nM T76685 CE1IJ5 71680722 Ki = 825 nM T76685 C14BYK 71680878 Ki > 10000 nM T76685 CY1ZL3 71680879 Ki > 10000 nM T76685 C2EMP9 71680880 Ki > 10000 nM T76685 C9ECU3 71680881 Ki > 10000 nM T76685 C3HR1X 71680882 Ki > 10000 nM T76685 C5AYI9 71681038 Ki > 10000 nM T76685 CQI90H 71681039 Ki > 10000 nM T76685 CFBR90 71681040 Ki > 10000 nM T76685 CVW58F 71681041 Ki > 10000 nM T76685 C0SOY4 71681042 Ki > 10000 nM T76685 C12PXS 71681193 Ki > 10000 nM T76685 C3KQZ0 71681194 Ki > 10000 nM T76685 C0S3LB 71681195 Ki > 10000 nM T76685 CY6AJ7 71681196 Ki > 10000 nM T76685 C5K9FS 71681197 Ki > 10000 nM T76685 CXC1Y5 71681346 Ki > 10000 nM T76685 CCO9K8 71681347 Ki > 10000 nM T76685 C6WQ9U 71681348 Ki > 10000 nM T76685 C3HUW6 71681349 Ki > 10000 nM T76685 C9LV4D 71681350 Ki > 10000 nM T76685 CVB7N1 71681500 Ki > 10000 nM T76685 C5D8CU 71681501 Ki > 10000 nM T76685 C0JVS9 71681502 Ki > 10000 nM T76685 CMWR71 71681503 Ki > 10000 nM T76685 CWQ86H 71681504 Ki > 10000 nM T76685 C6MKX3 71681665 Ki > 10000 nM T76685 CB63MS 71681666 Ki > 10000 nM T76685 CDJH76 71682490 Ki > 10000 nM T76685 C48BSN 71682637 Ki > 10000 nM T76685 C0O9HE 71682639 Ki = 3660 nM T76685 CZE6R2 71682640 Ki >= 10000 nM T76685 C2FBL9 71682641 Ki > 10000 nM T76685 CTOL05 71682642 Ki = 10000 nM T76685 CDX59H 71682795 Ki > 10000 nM T76685 C3S1OE 71682796 Ki = 7860 nM T76685 CNM1Y8 71682797 Ki >= 10000 nM T76685 C0HS4I 71682799 Ki = 613 nM T76685 C12BCL 71682928 Ki = 1278 nM T76685 CK0Y3J 71682950 Ki = 10200 nM T76685 C1AI4R 71683077 Ki = 527 nM T76685 CHZ86D 71683078 Ki = 1118 nM T76685 C2WK8I 71683079 Ki = 3290 nM T76685 C9RZG6 71683080 Ki = 2432 nM T76685 CGFD28 71683081 Ki = 420 nM T76685 C7WYZ1 71683082 Ki = 200 nM T76685 CUZ0W2 71717393 Ki = 1050 nM T76685 CM9RY4 71719542 EC50 > 10000 nM T76685 C1E9DF 71720136 EC50 > 10000 nM T76685 C1FYA8 71720426 EC50 = 32 nM T76685 C87UKF 71761847 EC50 = 12200 nM T76685 COW3E7 71762083 EC50 > 100000 nM T76685 C5BMG6 71764824 EC50 > 100000 nM T76685 CRFW13 71769176 Ki > 3000 nM T76685 CEND89 71769178 Ki > 1000 nM T76685 CLH7R3 71769179 Ki > 3000 nM T76685 C9MGJ3 71769180 Ki > 3000 nM T76685 CM14GO 71769181 Ki > 3000 nM T76685 CV2ZY6 71769306 Ki > 3000 nM T76685 C7KC5H 71769416 Ki > 1000 nM T76685 C58UGJ 71769417 Ki > 1000 nM T76685 C0UEZ7 71769418 Ki > 3000 nM T76685 CXHB14 71769420 Ki > 3000 nM T76685 C6S8AW 71769535 Ki > 3000 nM T76685 CS61FU 71819307 EC50 = 18 nM T76685 CBK6T9 72546989 IC50 = 8600 nM T76685 CJEP26 72696921 IC50 > 1000 nM T76685 CX9S4J 72696925 IC50 > 1000 nM T76685 CV0A9W 72697216 IC50 > 1000 nM T76685 C3GZO0 72697217 IC50 > 1000 nM T76685 CM6E8A 72697363 IC50 > 1000 nM T76685 C0ELS4 72713000 Ki = 2.55 nM T76685 CIA04R 72713195 Ki = 3.35 nM T76685 C4GL6T 72713198 Ki = 4.01 nM T76685 C41DNA 72713406 Ki = 2.67 nM T76685 C1Z8XN 72713407 Ki = 2.02 nM T76685 CLO9N1 72713633 Ki = 6.1 nM T76685 CT8GI1 72714379 EC50 > 10000 nM T76685 C5Z7JD 72714381 IC50 > 10000 nM T76685 COS7P3 72714471 IC50 > 10000 nM T76685 C5UDE2 72714472 IC50 > 10000 nM T76685 C1ULX5 72714474 EC50 > 10000 nM T76685 CPCW35 72714476 IC50 > 10000 nM T76685 C6O0TP 72714569 EC50 > 10000 nM T76685 CZHT65 72714571 IC50 > 10000 nM T76685 CN21QZ 72715287 EC50 > 10000 nM T76685 C1UVK7 72715369 EC50 > 10000 nM T76685 CG76DM 72715370 IC50 > 10000 nM T76685 CTY74C 72715372 EC50 > 10000 nM T76685 CWZ3M4 72715374 EC50 > 10000 nM T76685 C86BMU 72715375 EC50 > 10000 nM T76685 C1OHD4 72715447 IC50 > 10000 nM T76685 CJHR59 72715448 IC50 > 10000 nM T76685 CYPK25 72715612 EC50 > 10000 nM T76685 C5PL4U 72715613 EC50 > 10000 nM T76685 CZ5G1H 72715614 EC50 > 10000 nM T76685 CSBN82 72715615 EC50 > 10000 nM T76685 C4XTS1 72715697 EC50 > 10000 nM T76685 C8WQS4 72792900 Ki = 10 nM T76685 C58FDW 72792964 Ki = 4000 nM T76685 C6ZG1U 72792965 Ki = 4.2 nM T76685 C6JH0N 72792966 Ki = 29 nM T76685 CBM7W0 72793032 Ki = 28 nM T76685 CNHI43 72793033 Ki = 9 nM T76685 C5E7IF 72793034 Ki = 15 nM T76685 CR4U6G 72793098 Ki = 8.4 nM T76685 CX38EH 72793099 Ki = 1.4 nM T76685 CNV1J0 72793100 Ki = 3 nM T76685 CIT58M 72793169 Ki = 1.6 nM T76685 CUDY26 72793170 Ki = 1.9 nM T76685 CK01EC 72793171 Ki = 1.7 nM T76685 C72LSF 72793172 Ki = 12 nM T76685 CJ5YG1 72793173 Ki = 2.9 nM T76685 C2G7FX 72793239 Ki = 5 nM T76685 C1XR0U 72793240 Ki = 5 nM T76685 CNFA68 72793323 Ki = 3.2 nM T76685 CHW6N1 72793324 Ki = 92 nM T76685 C8G0MY 72793393 Ki = 77 nM T76685 C7B2VP 72941840 Ki = 1.259 nM T76685 CUA89W 72946872 IC50 = 180 nM T76685 C6F2UL 72948233 Ki = 134 nM T76685 CO5A1Z 72948234 Ki = 454 nM T76685 C7BCR9 72948235 Ki = 2603 nM T76685 C3Z2QA 72948236 Ki = 747 nM T76685 C68ASV 72948423 Ki = 1469 nM T76685 C6VRG9 72948424 Ki = 20.2 nM T76685 C3T0EL 72948425 Ki > 10000 nM T76685 CMF3P1 72948426 Ki = 52.4 nM T76685 C5Y8KP 72948428 Ki = 115 nM T76685 CTMP71 72948605 Ki = 96.6 nM T76685 C9WB7A 72948606 Ki = 127 nM T76685 C9POG2 72948607 Ki = 5.71 nM T76685 C9VFH8 72948608 Ki = 6.5 nM T76685 C91XBO 72948609 Ki = 9.85 nM T76685 C0MJ4P 72948610 Ki = 2.35 nM T76685 CI43RQ 72948611 Ki = 3.62 nM T76685 C9QMP3 72948786 Ki = 2.55 nM T76685 C1YL7A 72948787 Ki = 237 nM T76685 CWC76H 72950702 Ki = 0.859 nM T76685 CFID82 72950851 Ki = 8520 nM T76685 C27BSA 72950872 Ki = 1.18 nM T76685 C7U5EY 72950873 Ki = 15.9 nM T76685 CW87VS 72950874 Ki = 22.9 nM T76685 CB1K7N 72950875 Ki = 23.3 nM T76685 CH6TB0 72950876 Ki = 82.9 nM T76685 CW83DK 73213196 Ki > 10000 nM T76685 CX1H7E 73346065 Ki > 1000 nM T76685 C9JT1Q 73353637 Ki = 8670 nM T76685 CALG02 73354922 Ki = 12.2 nM T76685 C2E7QW 75201901 IC50 = 2100 nM T76685 C67UZL 76285447 Ki = 530 nM T76685 CV32SE 76309966 EC50 > 100000 nM T76685 C7T4EN 76310302 Ki > 10000 nM T76685 C0XBS8 76310303 Ki = 1830 nM T76685 CRDT21 76310304 Ki = 208 nM T76685 CUKW03 76310494 Ki > 10000 nM T76685 CWP1I7 76310495 Ki = 70 nM T76685 C70IVL 76310496 Ki = 23 nM T76685 CZCX06 76310497 Ki = 63 nM T76685 C2REF3 76310520 Ki = 24.8 nM T76685 C1JRI4 76310521 Ki = 3093 nM T76685 CG3D6K 76310535 EC50 > 17000 nM T76685 CV13PU 76310709 Ki = 3800 nM T76685 CK2XF6 76310722 IC50 = 222 nM T76685 C0BU4W 76310723 IC50 = 2280 nM T76685 C1ORB8 76310724 IC50 = 878 nM T76685 C0GPH6 76313156 Ki = 31.1 nM T76685 CQR92A 76313974 Ki > 8000 nM T76685 CH8K9Z 76313975 Ki = 563 nM T76685 CHKE18 76313976 Ki = 186 nM T76685 CKJ58T 76314156 Ki > 10000 nM T76685 C4C3HN 76314157 Ki = 243 nM T76685 CT9X1Q 76314180 Ki = 55 nM T76685 C0X5AU 76314195 EC50 > 17000 nM T76685 CI38KM 76314347 IC50 = 17800 nM T76685 CVSF70 76316704 Ki = 18.2 nM T76685 CSL9B8 76317193 EC50 = 948 nM T76685 CIJ3R1 76317524 Ki > 7000 nM T76685 CNH7R5 76317725 Ki = 8.8 nM T76685 C7NL6Z 76317738 Ki = 24 nM T76685 C8R9KD 76317739 Ki = 1270 nM T76685 CVI1O0 76317755 EC50 = 913 nM T76685 CRF6T0 76317756 EC50 > 17000 nM T76685 C1YVQ3 76317757 EC50 > 17000 nM T76685 CGI2O5 76317912 Ki = 2600 nM T76685 C1I2UO 76317913 Ki = 1400 nM T76685 CE5M1O 76317914 Ki > 10000 nM T76685 CQC2I9 76317932 IC50 = 8440 nM T76685 CY8Q4O 76317933 IC50 = 2100 nM T76685 CG1N4V 76317934 IC50 = 947 nM T76685 CO4IL2 76317959 Ki = 10600 nM T76685 CPF5Y0 76320912 Ki = 79 nM T76685 CRPD48 76321243 Ki = 129 nM T76685 C1L5EW 76321244 Ki > 5000 nM T76685 C8S1FB 76321458 EC50 > 17000 nM T76685 C04ELZ 76321459 EC50 > 17000 nM T76685 CO5LP6 76321460 EC50 > 17000 nM T76685 CI2F6O 76321461 EC50 = 123 nM T76685 C20OWQ 76321462 EC50 > 17000 nM T76685 C4M8ZY 76321622 Ki = 200 nM T76685 CSXH87 76321623 Ki = 3000 nM T76685 CO05BZ 76321641 IC50 = 3750 nM T76685 CLS36H 76321951 Ki = 3170 nM T76685 CXW8I6 76324059 Ki = 100 nM T76685 CRV4F9 76324060 Ki = 399.9 nM T76685 CMP3Z8 76324864 Ki > 10000 nM T76685 CX2F4H 76325028 Ki > 10000 nM T76685 CBLG65 76325060 EC50 > 17000 nM T76685 CE3YU9 76325061 EC50 > 17000 nM T76685 C3NB1K 76325062 EC50 > 17000 nM T76685 C0HA3K 76325063 EC50 > 17000 nM T76685 CFBZ86 76325097 Ki = 810 nM T76685 C1W8HB 76325234 Ki = 560 nM T76685 CO05NW 76325235 Ki = 11000 nM T76685 CR2LF5 76325256 IC50 = 388 nM T76685 C5GI9Z 76325292 Ki > 10000 nM T76685 CN4D3M 76328423 Ki = 25.8 nM T76685 CSQ0H6 76328424 Ki = 190 nM T76685 CFGB61 76328601 Ki = 1830 nM T76685 CWIF86 76328602 Ki > 10000 nM T76685 CI0SB5 76328619 Ki > 10000 nM T76685 C91YWU 76328633 EC50 > 17000 nM T76685 C3BZ6H 76328634 EC50 > 17000 nM T76685 C1LN2I 76328635 EC50 > 17000 nM T76685 CX31IO 76328636 EC50 > 17000 nM T76685 C5AV9G 76328789 Ki > 40000 nM T76685 C4QH5I 76328790 Ki > 40000 nM T76685 C30AMV 76328791 Ki > 40000 nM T76685 CB1KJ6 76328792 Ki = 1300 nM T76685 C7GD9E 76331283 Ki = 327.3 nM T76685 CC56VG 76331284 Ki = 19.8 nM T76685 CWD5R4 76331595 IC50 = 345 nM T76685 CR6IJ1 76331611 Ki = 14180 nM T76685 CPV9G7 76331637 IC50 = 41 nM T76685 CBE63L 76331817 Ki > 10000 nM T76685 CK20OT 76332105 Ki = 1900 nM T76685 CDUQ61 76332106 Ki = 247 nM T76685 CHV15W 76332282 Ki = 1623 nM T76685 CU4B7F 76332298 Ki = 24 nM T76685 CT5GH7 76332299 Ki = 1920 nM T76685 C9H2JW 76332300 Ki = 884 nM T76685 CTDG64 76332315 EC50 > 17000 nM T76685 C6CI5P 76332316 EC50 > 17000 nM T76685 CPET62 76334865 Ki = 256.4 nM T76685 CA1N6F 76334866 Ki = 11.67 nM T76685 C4H1UV 76334867 Ki = 240.99 nM T76685 CJD08P 76335394 EC50 > 100000 nM T76685 CHRV01 76335726 Ki = 66.4 nM T76685 C73ZEL 76335925 Ki > 10000 nM T76685 CSF2G0 76335926 Ki = 35 nM T76685 C8ZW2C 76335938 Ki = 2734 nM T76685 CFP9L2 76335946 EC50 > 17000 nM T76685 CTG51J 76336093 Ki > 10000 nM T76685 CBVR96 76336107 IC50 = 1840 nM T76685 CHI98A 76336108 IC50 = 4730 nM T76685 C6DA9V 77529583 Ki = 2300 nM T76685 CW08SU 78320048 IC50 = 120 nM T76685 C48YMX 84382039 Ki > 10000 nM T76685 CQE10H 85468767 Ki > 10000 nM T76685 CA0Y8G 85469571 Ki > 10000 nM T76685 CQ9H4U 86277844 IC50 > 10000 nM T76685 CYR30A 86625327 Ki = 0.1259 nM T76685 C98LWE 86669644 EC50 = 86 nM T76685 CW3TR2 86669645 EC50 = 19.1 nM T76685 C6ZWO8 86669647 EC50 = 51 nM T76685 CU98CB 86669673 EC50 = 297 nM T76685 CBP12Z 86688562 EC50 = 15.6 nM T76685 C5PLO7 86688563 EC50 > 30000 nM T76685 CISP51 86688570 EC50 > 30000 nM T76685 CDX5N1 87700872 Ki = 0.1 nM T76685 CIW56T 88530818 EC50 = 17000 nM T76685 CV82BP 88530819 EC50 > 20000 nM T76685 CMO84Z 88924517 IC50 > 10000 nM T76685 CY5MX1 89044257 EC50 > 20000 nM T76685 C6WZH9 89044294 EC50 > 20000 nM T76685 CO7J6V 90054857 Ki = 107 nM T76685 C2HLG9 90654966 Ki = 5055 nM T76685 CBG40L 90654968 EC50 > 10000 nM T76685 CV05HR 90654970 EC50 > 1.5 nM T76685 CHN43D 90654972 EC50 > 50000 nM T76685 CVY83X 90667465 Ki > 10000 nM T76685 C85BUR 90667466 Ki > 10000 nM T76685 C0FZU2 90667467 Ki > 10000 nM T76685 C4MF8A 90667653 Ki > 10000 nM T76685 CR2WI4 90667654 Ki > 10000 nM T76685 C8N0LA 90667655 Ki > 10000 nM T76685 CU23VX 90667656 Ki = 2090 nM T76685 CR8I5E 90667657 Ki > 10000 nM T76685 CI61LD 90667658 Ki > 10000 nM T76685 C7P2EG 90667659 Ki > 10000 nM T76685 CS5DZ4 90667660 Ki = 2130 nM T76685 C31ZMH 90667661 Ki = 2160 nM T76685 CT37YL 90667662 Ki = 2290 nM T76685 CJ7V0Y 90667663 Ki = 850 nM T76685 C54BTS 90667664 Ki > 10000 nM T76685 CJP21Z 90667665 Ki > 10000 nM T76685 C9RM7U 90667666 Ki > 10000 nM T76685 CB5VS3 91755003 EC50 = 1620 nM T76685 CWS6G3 91824816 Ki > 40000 nM T76685 CL7S4U 91844670 EC50 = 8.2 nM T76685 C0Z5LH 91936927 EC50 = 2.1 nM T76685 C1MB3D 92279023 Ki > 10000 nM T76685 C5J8EZ 101609852 Ki > 10000 nM T76685 CQS1P5 101882735 Ki = 96.1 nM T76685 CHSE20 101882736 Ki = 750 nM T76685 C7IP2A 101882737 Ki > 10000 nM T76685 C0G8PM 101884092 Ki = 1084 nM T76685 C1FMO9 101884564 Ki > 10000 nM T76685 C9ED8P 101884565 Ki > 10000 nM T76685 CHQ86Y 101884566 Ki > 10000 nM T76685 CAM2R6 101884567 Ki > 10000 nM T76685 C5P8CV 101884568 Ki > 10000 nM T76685 CX08DR 101884569 Ki > 10000 nM T76685 C0CB8R 101884572 Ki > 10000 nM T76685 CNA2H8 101884573 IC50 > 10000 nM T76685 CLYG63 101884574 IC50 > 10000 nM T76685 CF1D6S 101898797 Ki = 7.22 nM T76685 C2POM8 101898798 Ki > 10000 nM T76685 CH3ZJ1 102339340 Ki = 470 nM T76685 C58ZBN 102506267 Ki = 31 nM T76685 CEM4P9 102506268 Ki = 830 nM T76685 CQF3M5 102514739 Ki > 3000 nM T76685 COF7T3 109112982 EC50 > 10000 nM T76685 CYT61B 117698842 EC50 > 20000 nM T76685 C5BWP4 117910962 IC50 > 10000 nM T76685 CSG6E5 117911325 IC50 = 203 nM T76685 C4M9RG 117911437 IC50 = 228 nM T76685 C56JSF 117911440 IC50 > 10000 nM T76685 CRPJ57 117911450 IC50 > 10000 nM T76685 CF94VY 117911451 IC50 = 166 nM T76685 CL8CT9 117911478 IC50 = 888 nM T76685 CM1YP7 117911495 IC50 = 189 nM T76685 CWNB39 117911505 EC50 = 209 nM T76685 CFNT01 117911520 EC50 = 207 nM T76685 C41NLJ 117911680 EC50 = 43 nM T76685 C8I4SP 117923246 EC50 = 64 nM T76685 CTQ57B 117923262 EC50 = 28.2 nM T76685 CA8EP5 117923263 EC50 = 683 nM T76685 C0P6TC 117923264 EC50 = 28.2 nM T76685 C3YSH0 118323940 EC50 = 122 nM T76685 C1Z9RI 118323944 EC50 = 399 nM T76685 CS6A0V 118323946 EC50 = 10.8 nM T76685 CO1I2G 118323957 EC50 = 220 nM T76685 CP19AD 118323960 EC50 = 310 nM T76685 C4ANZ8 118323971 EC50 = 108 nM T76685 CF0BH7 118323974 EC50 = 290 nM T76685 CDT29M 118323979 EC50 = 1100 nM T76685 C1TDN2 118323981 EC50 = 144 nM T76685 C0HAR6 118323983 EC50 = 121 nM T76685 CCL1H8 118323989 EC50 = 8.4 nM T76685 CKN63V 118323997 EC50 = 6 nM T76685 COH45S 118323999 EC50 = 228 nM T76685 CN4E6J 118324004 EC50 = 51 nM T76685 C5JAE7 118324005 EC50 = 157 nM T76685 CU6IQ3 118324016 EC50 = 159 nM T76685 CQC1A2 118324032 EC50 = 1550 nM T76685 C3R9TY 118324047 EC50 = 15 nM T76685 CP8Q3X 118324048 EC50 = 604 nM T76685 CB0IA3 118324050 EC50 = 269 nM T76685 CF1MC2 118324059 EC50 = 24 nM T76685 CSEF20 118324060 EC50 = 10.9 nM T76685 C7AO1M 118324066 EC50 = 396 nM T76685 CQ67PB 118324068 EC50 = 817 nM T76685 C3KYS6 118324079 EC50 = 625 nM T76685 CC2KB9 118324098 EC50 = 438 nM T76685 CMHK20 118324101 EC50 = 876 nM T76685 CQ7A3N 118324116 EC50 = 94.4 nM T76685 CT6GJ1 118324120 EC50 = 13 nM T76685 CC7F2I 118324123 EC50 = 20.4 nM T76685 C6EZ9B 118324131 EC50 = 22 nM T76685 CQH25F 118324141 EC50 = 14 nM T76685 C8L0YE 118324167 Ki > 10000 nM T76685 CZ09WH 118324183 Ki = 4.38 nM T76685 CCU41D 118324204 Ki = 4174 nM T76685 CW91NY 118324233 Ki = 4083 nM T76685 CD1Q0F 118329953 EC50 = 4140 nM T76685 C1EF7O 118329959 EC50 = 1210 nM T76685 CS79MQ 118329962 EC50 = 204 nM T76685 CIRF81 118329963 EC50 = 2330 nM T76685 CS3QP9 118329966 EC50 = 75 nM T76685 CWD7H3 118329970 EC50 = 10 nM T76685 C0N7BQ 118329972 EC50 = 29 nM T76685 CE3DI2 118329973 EC50 = 64.2 nM T76685 CTX50R 118329986 EC50 = 13.5 nM T76685 CQD27U 118329991 EC50 = 9700 nM T76685 CLQ6D2 118329993 EC50 = 1284 nM T76685 CE30FQ 118329995 EC50 = 92 nM T76685 CX7HP5 118332418 Ki = 149 nM T76685 CW0KL9 118332421 Ki = 607 nM T76685 C3IQ7F 118332422 Ki = 623 nM T76685 C62GQO 118332423 Ki = 647 nM T76685 CPY5T1 118332424 Ki = 1000 nM T76685 CUIG26 118332426 Ki = 862 nM T76685 CFTD05 118332428 Ki > 10000 nM T76685 CO0R9Z 118332431 Ki = 8528 nM T76685 CZ7C5S 118577928 Ki > 3000 nM T76685 C2TF0N 118577933 Ki > 3000 nM T76685 C0B3LV 118577936 Ki > 3000 nM T76685 CIJF40 118577937 Ki > 3000 nM T76685 CJ1HD0 118577940 Ki > 3000 nM T76685 CQK7V8 118577942 Ki > 3000 nM T76685 CW3C2E 118577959 Ki > 3000 nM T76685 CFUY17 118577977 Ki > 3000 nM T76685 CGL1Y4 118577980 Ki > 3000 nM T76685 CY3PA2 118643310 Ki > 10000 nM T76685 CTC9R6 118643314 Ki > 10000 nM T76685 C6CG5I 118643315 Ki > 10000 nM T76685 C3PQS9 118643388 Ki > 10000 nM T76685 C6E7PK 118643393 Ki > 10000 nM T76685 C6XYO1 118643396 Ki > 10000 nM T76685 CI2AP3 118643406 Ki > 10000 nM T76685 CIHQ76 118643434 Ki > 10000 nM T76685 C7X1ZB 118706308 EC50 = 1348.96 nM T76685 CC2G6V 118706310 EC50 = 25118.86 nM T76685 CFL1Z4 118706312 EC50 = 6309.57 nM T76685 C6SD4K 118706313 EC50 = 34673.69 nM T76685 CQ9B4G 118706315 EC50 = 23988.33 nM T76685 C16JGM 118706317 EC50 = 25703.96 nM T76685 CZ24EM 118706318 EC50 = 17378.01 nM T76685 CN4G2U 118707905 Ki = 8600 nM T76685 CUS4F2 118707906 Ki > 20000 nM T76685 CI23QP 118707907 Ki = 310 nM T76685 C0ABJ8 118709741 Ki = 1240 nM T76685 C9AO5K 118709742 Ki = 2080 nM T76685 CF6CR0 118709743 Ki = 830 nM T76685 C5D4LR 118710063 EC50 = 2818.38 nM T76685 C1C6JD 118710064 EC50 = 112 nM T76685 CYO84T 118710065 EC50 = 3850 nM T76685 CTOF52 118710153 EC50 = 15000 nM T76685 C6UPI9 118710154 EC50 = 40700 nM T76685 C5LMQ9 118710155 EC50 = 9549.93 nM T76685 CKJX93 118710156 EC50 = 8709.64 nM T76685 CC57ZA 118710157 EC50 = 13489.63 nM T76685 CQ1L3K 118710158 EC50 = 8511.38 nM T76685 CAET43 118710159 EC50 = 7585.78 nM T76685 CS8C4L 118710160 EC50 = 23988.33 nM T76685 CQ92ZT 118710161 EC50 = 3160 nM T76685 CJ9P7E 118710162 EC50 = 10471.29 nM T76685 CO48YL 118710164 EC50 = 16218.1 nM T76685 CR4G6U 118710165 EC50 = 7240 nM T76685 C98RHP 118710166 EC50 = 8850 nM T76685 C0VP2R 118710167 EC50 = 2950 nM T76685 CYEB75 118710168 EC50 = 776 nM T76685 CS0U7R 118710169 EC50 = 501 nM T76685 CVC6T1 118710170 EC50 = 109.65 nM T76685 CTOP59 118710171 EC50 = 1096.48 nM T76685 CP7AZ2 118710172 EC50 = 660.69 nM T76685 CIQ9L8 118710173 EC50 = 123 nM T76685 C9AZU0 118710175 EC50 = 1905.46 nM T76685 CSP5J3 118710952 Ki = 12.8 nM T76685 C9CM3X 118710953 Ki = 264.4 nM T76685 CW5S6I 118710954 Ki = 17.2 nM T76685 CW15QT 118710955 Ki = 132.2 nM T76685 CD1A3B 118710956 Ki > 10000 nM T76685 CV9Q4L 118710957 Ki = 177.8 nM T76685 CT12DE 118710958 Ki = 1890 nM T76685 CE3LG5 118710959 Ki > 10000 nM T76685 CRVG42 118710960 Ki > 10000 nM T76685 CK8C0R 118710961 Ki = 136.3 nM T76685 CCIE15 118710962 Ki = 438 nM T76685 C0CS2E 118710963 Ki = 397 nM T76685 CJ35MC 118710964 Ki > 10000 nM T76685 C4WUB9 118710965 Ki > 10000 nM T76685 C37ZAO 118710966 Ki > 10000 nM T76685 C89QBL 118710967 Ki > 10000 nM T76685 CRDH69 118710968 Ki > 10000 nM T76685 C6CP7G 118710969 Ki > 10000 nM T76685 CSE1V9 118710970 Ki = 845.5 nM T76685 CW09BI 118710971 Ki = 1782 nM T76685 CB8SV3 118710972 Ki = 2770 nM T76685 CM91UF 118710973 Ki = 2070 nM T76685 C9S5DN 118710974 Ki = 900 nM T76685 CAK1P8 118710975 Ki > 10000 nM T76685 CI9NB6 118710976 Ki = 1060 nM T76685 CYGH30 118710977 Ki = 1140 nM T76685 CJ7UB1 118711121 Ki > 10000 nM T76685 CQU6G8 118711283 Ki = 10000 nM T76685 CA6F4R 118711284 Ki > 10000 nM T76685 CIH8W4 118712416 Ki > 10000 nM T76685 CD5U3M 118712417 Ki > 10000 nM T76685 CRML68 118712418 Ki > 10000 nM T76685 CHD54U 118712419 Ki = 2100 nM T76685 COV62X 118712420 Ki = 1100 nM T76685 CA3HS1 118712421 Ki > 10000 nM T76685 C4C9AZ 118712672 Ki > 10000 nM T76685 CS76HN 118712673 Ki > 10000 nM T76685 CUV5Y0 118715454 EC50 > 30000 nM T76685 CP41KA 118716098 IC50 = 27.4 nM T76685 C6GI9U 118716099 IC50 = 125 nM T76685 C0C7KH 118716100 IC50 = 372 nM T76685 CLXF54 118716101 IC50 = 693 nM T76685 C8SMJ6 118716102 IC50 = 317 nM T76685 C0ZH6P 118716103 IC50 = 181 nM T76685 CUP13J 118716104 IC50 = 311 nM T76685 CG08CE 118716105 EC50 = 1520 nM T76685 CT75ZN 118716106 IC50 = 867 nM T76685 CI9K5X 118716107 IC50 = 1360 nM T76685 C6F7MO 118716108 IC50 = 501 nM T76685 CK2V3X 118716109 IC50 = 53.7 nM T76685 CXTP42 118716110 IC50 = 156 nM T76685 CH6EQ5 118716111 IC50 = 104 nM T76685 CI51GD 118716112 IC50 = 251 nM T76685 C5I7EF 118716113 IC50 = 98 nM T76685 CN4QJ1 118716114 IC50 = 33 nM T76685 CCMZ95 118716115 IC50 = 100 nM T76685 C41GVI 118716116 IC50 = 1640 nM T76685 CI98FK 118716117 IC50 = 312 nM T76685 CWL0K7 118716118 IC50 > 10000 nM T76685 CQW4C7 118716119 IC50 = 1880 nM T76685 C6T1HF 118716120 IC50 > 10000 nM T76685 CH7C4E 118716121 IC50 = 161 nM T76685 C9OJX0 118716122 IC50 = 716 nM T76685 CD4G6H 118716123 IC50 = 135 nM T76685 C8ZAG3 118716124 Ki = 9 nM T76685 CI76QT 118717840 EC50 > 3162.28 nM T76685 CDO6U3 118717842 EC50 = 251.19 nM T76685 CMIL98 118717845 EC50 = 1584.89 nM T76685 CQJ98W 118717846 EC50 = 1000 nM T76685 C7HOR2 118717847 EC50 = 316.23 nM T76685 C6SIV2 118717852 EC50 = 100 nM T76685 CJZ70E 118717859 EC50 = 501.19 nM T76685 CXL7H2 118717860 EC50 = 794.33 nM T76685 C4BI7A 118717874 EC50 = 794.33 nM T76685 CE0Y1A 118717875 EC50 > 3162.28 nM T76685 CQ4CD8 118717885 EC50 = 63.1 nM T76685 CW6OU8 118717886 EC50 > 3162.28 nM T76685 C0Y2PI 118717887 EC50 > 3162.28 nM T76685 C9DY8C 118717888 EC50 = 630.96 nM T76685 CRE04K 118717899 EC50 = 501.19 nM T76685 CH9PX5 118717900 EC50 = 316.23 nM T76685 C1J3NW 118717902 EC50 = 251.19 nM T76685 C5K3IG 118717904 EC50 = 39.81 nM T76685 CKZ72N 118717906 EC50 = 10 nM T76685 CNP6Z8 118717911 EC50 > 3162.28 nM T76685 CNU15K 118717912 EC50 = 125.89 nM T76685 CT3K7J 118717913 EC50 = 125.89 nM T76685 CON02E 118717918 Ki = 1.259 nM T76685 C8YJB0 118717920 EC50 = 158.49 nM T76685 C3G4XO 118717935 EC50 = 501.19 nM T76685 C6KQT7 118717936 EC50 = 1258.93 nM T76685 C9VPN4 118717937 EC50 = 1995.26 nM T76685 C3XP4F 118719586 Ki = 2314 nM T76685 CKXB38 118719587 Ki = 908 nM T76685 CVW1U3 118719588 Ki > 10000 nM T76685 C3ZD9J 118719589 Ki > 10000 nM T76685 CUF2I9 118719590 Ki > 10000 nM T76685 CZDV38 118719591 Ki > 10000 nM T76685 C46ZPY 118719592 Ki > 10000 nM T76685 CO4BY2 118719593 Ki > 10000 nM T76685 CJ3N1Q 118719594 Ki > 10000 nM T76685 CUC56R 118719595 Ki > 10000 nM T76685 CIAP43 118719596 Ki > 10000 nM T76685 CZJ47G 118719597 Ki > 10000 nM T76685 CWJ26O 118719598 Ki > 10000 nM T76685 CX3UG7 118719599 Ki = 1011 nM T76685 C8BYZ5 118719600 Ki = 22.59 nM T76685 CXJA89 118719601 Ki = 35.67 nM T76685 C4YA1O 118719602 Ki = 3262 nM T76685 C40MOC 118719603 Ki = 430 nM T76685 CW0L8Y 118719604 Ki > 10000 nM T76685 C5LA2D 118719605 Ki = 3444 nM T76685 CPK5M3 118719606 Ki = 32.7 nM T76685 C1NWH9 118719607 Ki = 66.7 nM T76685 C1PD4O 118719608 Ki = 52.9 nM T76685 CDW0B1 118720256 EC50 > 20000 nM T76685 C05YAJ 118720257 EC50 > 20000 nM T76685 C96TEL 118720552 EC50 = 7.4 nM T76685 C9X6JL 118720553 EC50 = 2.1 nM T76685 CRW5A6 118720554 EC50 = 4.4 nM T76685 C4DJ0Z 118720555 EC50 = 0.3 nM T76685 CSF28U 118720556 EC50 = 21.7 nM T76685 CA2Q0R 118720557 EC50 = 381 nM T76685 C17YFC 118720558 EC50 = 341 nM T76685 CH0A5R 118720559 EC50 > 30000 nM T76685 CH0AS9 118720560 EC50 = 1300 nM T76685 C2AW1O 118720561 EC50 > 30000 nM T76685 C74UHD 118720562 EC50 = 43 nM T76685 CN42VO 118720563 EC50 = 3400 nM T76685 C6ZT3W 118720564 EC50 > 30000 nM T76685 CY6T4M 118720565 EC50 = 105 nM T76685 CK8V5U 118720566 EC50 > 30000 nM T76685 C6FDB2 118720567 EC50 > 30000 nM T76685 CP80QJ 118720568 EC50 > 30000 nM T76685 CWTU50 118720569 EC50 > 30000 nM T76685 CI3O6C 118720570 EC50 > 30000 nM T76685 C6XN4L 118720571 EC50 = 217 nM T76685 CDM1K3 118720572 EC50 > 30000 nM T76685 CR6VQ9 118720573 EC50 > 30000 nM T76685 C5OHY6 118720574 EC50 > 30000 nM T76685 C2TG4E 118720575 EC50 > 30000 nM T76685 C42GIB 118720576 EC50 > 30000 nM T76685 CMIB62 118720577 EC50 > 30000 nM T76685 C0MXK9 118720578 EC50 > 30000 nM T76685 CGH7U9 118720579 EC50 > 30000 nM T76685 C9SJH4 118720580 EC50 > 30000 nM T76685 C0U8PC 118720581 EC50 = 3600 nM T76685 CRZK09 118720582 EC50 > 30000 nM T76685 C62GLY 118720583 EC50 > 30000 nM T76685 CPB17U 118720584 EC50 > 30000 nM T76685 C2EDL9 118722126 EC50 > 100000 nM T76685 CNRL68 118722145 EC50 = 1600 nM T76685 CYP8S3 118722147 EC50 = 2800 nM T76685 CZ0R3B 118722156 EC50 > 25000 nM T76685 CM3YE9 118722157 EC50 = 16000 nM T76685 CLS38E 118722158 EC50 > 25000 nM T76685 CR2E1P 118722159 EC50 > 25000 nM T76685 C4A9RF 118722160 EC50 = 10000 nM T76685 CTND40 118722161 EC50 > 25000 nM T76685 CBCN25 118722162 EC50 > 25000 nM T76685 CS6CX9 118726686 Ki > 10000 nM T76685 C3O6VM 118726687 Ki > 10000 nM T76685 CTW1E4 118726688 Ki = 656 nM T76685 CU2XS4 118726689 Ki = 1090 nM T76685 CZS7Q0 118726769 Ki = 160 nM T76685 C2CZ9R 118726770 Ki = 180 nM T76685 C4U0TC 118726771 Ki = 1494 nM T76685 CBG38P 118726772 Ki = 1550 nM T76685 C87AZE 118727849 IC50 = 483 nM T76685 CN5DV2 118727850 IC50 = 1800 nM T76685 CU6T1D 118727851 IC50 = 3620 nM T76685 CDXC42 118727852 IC50 > 10000 nM T76685 CE1T0M 118727853 IC50 > 10000 nM T76685 CMD62P 118727854 IC50 > 10000 nM T76685 CWB01A 118727855 IC50 > 10000 nM T76685 CM5D8T 118727856 IC50 = 3150 nM T76685 CG0CI1 118727857 IC50 = 2560 nM T76685 C8G9LQ 118727858 IC50 = 2430 nM T76685 CPS6Q0 118728139 EC50 = 1000 nM T76685 CV8YP1 118728142 EC50 = 253 nM T76685 CDNO97 118728581 IC50 = 5810 nM T76685 C6KO8C 118728582 IC50 = 831 nM T76685 CC3VS2 118728583 IC50 = 2100 nM T76685 C7N8LA 118728584 IC50 > 10000 nM T76685 C2ZAO7 118728585 IC50 > 10000 nM T76685 C9QJV2 118728586 IC50 = 2170 nM T76685 C6C1PD 118728587 IC50 = 4320 nM T76685 CH60QT 118728588 IC50 > 10000 nM T76685 CWO9C0 118728589 IC50 > 10000 nM T76685 CAJ0K3 118728590 IC50 > 10000 nM T76685 CP3I2H 118728591 IC50 = 361 nM T76685 C6WXP8 118728592 IC50 = 151 nM T76685 CH72RQ 118728593 IC50 = 318 nM T76685 CTY17R 118728594 IC50 = 79 nM T76685 C65PBY 118728595 IC50 = 605 nM T76685 C4CZH7 118728596 IC50 = 279 nM T76685 C0J8VB 118728597 IC50 = 319 nM T76685 CBDX93 118731518 Ki > 10000 nM T76685 C7CIR8 118731519 Ki = 4772 nM T76685 C3BMI7 118732560 EC50 > 10000 nM T76685 C29RBK 118732561 EC50 > 10000 nM T76685 CPY68L 118732562 EC50 > 10000 nM T76685 C9LR2Z 118732563 EC50 > 10000 nM T76685 CWYR05 118732564 EC50 > 10000 nM T76685 C5BUD9 118732565 EC50 > 10000 nM T76685 CCSR86 118732566 EC50 > 10000 nM T76685 C5OD3H 118732567 IC50 > 10000 nM T76685 CXI3Y5 118732568 IC50 > 10000 nM T76685 C7HPJ3 118732569 IC50 > 10000 nM T76685 C3FXW5 118732570 IC50 > 10000 nM T76685 CV52GQ 118732571 IC50 > 10000 nM T76685 CY31XU 118732572 IC50 > 10000 nM T76685 C12WUS 118732573 IC50 > 10000 nM T76685 CBL75P 118732574 IC50 > 10000 nM T76685 CUMB75 118732575 IC50 > 10000 nM T76685 C2MHZ6 118734857 Ki > 40000 nM T76685 C1IEC4 118734858 Ki > 40000 nM T76685 CA6R8C 118735104 Ki > 3000 nM T76685 CZK9S4 118735105 Ki > 3000 nM T76685 C9VBC6 118735106 Ki > 3000 nM T76685 CCZ36J 118735107 Ki > 3000 nM T76685 CH1N5T 118735108 Ki > 3000 nM T76685 CFLH28 118735109 Ki > 3000 nM T76685 C6BTX2 118735110 Ki > 3000 nM T76685 CNUC23 118735111 Ki > 3000 nM T76685 CV0RP2 118735112 Ki > 3000 nM T76685 CP21CI 118735884 Ki = 19.4 nM T76685 C14OKB 118735885 Ki = 800 nM T76685 C5T2XB 118735886 Ki = 2609 nM T76685 C89UAT 118735887 Ki = 551 nM T76685 C58TLB 118735888 Ki = 227 nM T76685 CB9CH4 118735889 Ki = 3761 nM T76685 CTC74N 118735890 Ki = 138.5 nM T76685 CK38BW 118735891 Ki = 630.3 nM T76685 CG6XJ8 118735892 Ki = 701.5 nM T76685 CPA03J 118735893 Ki > 10000 nM T76685 CN2VG3 118908760 EC50 = 301 nM T76685 CG3M8O 118908931 EC50 = 322 nM T76685 C8YKI5 118909030 EC50 > 10000 nM T76685 CX4PY8 121028259 EC50 > 10000 nM T76685 C7GH5N 121453184 EC50 = 2.09 nM T76685 C9QHM7 122180086 Ki = 117 nM T76685 CCY7M4 122180087 Ki = 224 nM T76685 C8Z6KE 122180088 Ki = 47 nM T76685 CQC97X 122181545 EC50 < 10000 nM T76685 C1MY7T 122182962 Ki > 10000 nM T76685 CX0D8H 122182963 Ki > 10000 nM T76685 CM9Z1Y 122182964 Ki > 10000 nM T76685 CTF89J 122182965 Ki > 10000 nM T76685 CL7FR1 122182966 Ki > 10000 nM T76685 CDUA90 122182967 Ki > 10000 nM T76685 CB3V2C 122182968 Ki > 10000 nM T76685 CN5H3A 122182969 Ki > 10000 nM T76685 C4HI6P 122182970 Ki > 10000 nM T76685 C9QDS4 122182971 Ki > 10000 nM T76685 C5CL4O 122182972 Ki > 10000 nM T76685 C1SVF8 122182973 Ki > 10000 nM T76685 CP8GV4 122182974 Ki > 10000 nM T76685 C9QMW0 122182975 Ki > 10000 nM T76685 C3I7FO 122182976 Ki > 10000 nM T76685 CXR07B 122183469 Ki = 590 nM T76685 CWP92F 122183470 Ki = 410 nM T76685 CO2P0J 122186206 Ki > 10000 nM T76685 CVA4X9 122186207 Ki = 298.6 nM T76685 CIMB95 122186208 Ki = 9429 nM T76685 C9M4RG 122186209 Ki > 10000 nM T76685 C6T7FD 122186210 Ki > 10000 nM T76685 C21IXD 122186211 EC50 > 5000 nM T76685 CI39PN 122186212 Ki = 4134 nM T76685 C1JKN9 122186213 Ki = 1138 nM T76685 CLYT85 122186214 Ki > 10000 nM T76685 C8SK3V 122186215 Ki > 10000 nM T76685 C3I6RX 122186216 Ki = 3326 nM T76685 C42KBM 122186217 Ki > 10000 nM T76685 CI0S8P 122186218 Ki = 2529 nM T76685 CPLO68 122186219 Ki > 10000 nM T76685 CL91KO 122186220 EC50 = 3280 nM T76685 C0B9OG 122186221 Ki > 10000 nM T76685 CEPZ53 122186222 Ki > 10000 nM T76685 CLXN43 122186223 EC50 = 2880 nM T76685 C4FA8H 122186224 Ki > 10000 nM T76685 CM1HG9 122186225 Ki > 10000 nM T76685 CYE3S0 122186226 Ki > 10000 nM T76685 CL7QJ3 122188721 Ki = 1470 nM T76685 C0Y7MH 122188723 Ki = 368 nM T76685 CL6ZK9 122188725 Ki > 5000 nM T76685 CY8A0I 122188726 Ki > 5000 nM T76685 CNOJ38 122188727 Ki > 5000 nM T76685 CM12WF 122188728 Ki > 5000 nM T76685 CZ5K3W 122188729 Ki > 5000 nM T76685 CN36ST 122188731 Ki > 5000 nM T76685 C0Y2HU 122188732 Ki = 3070 nM T76685 CY89ZL 122188733 Ki > 5000 nM T76685 CG8AB5 122188734 Ki > 5000 nM T76685 CASB97 122188735 Ki > 5000 nM T76685 C46EAN 122188736 Ki > 5000 nM T76685 CKPT42 122188737 Ki > 5000 nM T76685 C5SNP3 122188738 Ki > 5000 nM T76685 C5HC0Z 122188739 Ki > 5000 nM T76685 CPE05A 122188740 Ki > 5000 nM T76685 CDA10L 122366667 IC50 > 10000 nM T76685 C16IOX 123128346 IC50 = 6.8 nM T76685 C9JIL6 123233001 EC50 = 42.9 nM T76685 C3DWH0 123627357 EC50 = 1100 nM T76685 CUW54Z 123922722 EC50 > 10000 nM T76685 CDK95B 124021285 EC50 = 6100 nM T76685 CS9U3T 126502731 EC50 = 1500 nM T76685 CCQO62 126630141 EC50 = 56 nM T76685 CZ6G3E 126630168 EC50 = 457 nM T76685 C8CBI0 127026099 Ki = 8.82 nM T76685 CGFD26 127027049 Ki = 1.9 nM T76685 CYN8P2 127027323 Ki = 14.5 nM T76685 CIR76K 127027671 Ki = 44.4 nM T76685 C6E1TL 127027672 Ki = 9.6 nM T76685 CXK8J7 127027699 Ki = 28.9 nM T76685 CED8I2 127027701 Ki = 9.2 nM T76685 CO32AZ 127027987 Ki = 43.5 nM T76685 CM8VA4 127027989 Ki = 43 nM T76685 C4BY3G 127028018 Ki = 7.5 nM T76685 C18JNK 127029837 Ki > 40000 nM T76685 CZX4C2 127029838 Ki > 40000 nM T76685 C9FG1J 127029891 Ki > 10000 nM T76685 CT81PH 127029928 Ki > 40000 nM T76685 C39OXL 127029929 Ki > 10000 nM T76685 CY3LI1 127029930 Ki > 40000 nM T76685 C5SH7V 127030115 Ki > 10000 nM T76685 CN49LK 127030116 Ki > 40000 nM T76685 CV6Z5S 127030117 Ki > 10000 nM T76685 C1U2CM 127030118 Ki = 4033 nM T76685 C3L8GO 127030160 Ki > 40000 nM T76685 C3I4CH 127030161 Ki > 40000 nM T76685 CHMI58 127030184 Ki = 1852 nM T76685 CVDP63 127030185 Ki > 40000 nM T76685 CMO64X 127030260 Ki > 40000 nM T76685 CYBU18 127030261 Ki > 40000 nM T76685 C61MQJ 127030421 Ki > 10000 nM T76685 CN7A6R 127030422 Ki > 40000 nM T76685 CIMH58 127030534 Ki = 622 nM T76685 CXBY26 127030535 Ki = 488 nM T76685 CLRC71 127030536 Ki = 471 nM T76685 C4HSR6 127030537 Ki = 3214 nM T76685 C2NVB3 127030843 Ki = 717 nM T76685 C4WXA8 127030844 Ki = 2483 nM T76685 C9F2UM 127030845 Ki = 653 nM T76685 C3Y6ZT 127031443 Ki > 10000 nM T76685 CTE32L 127031950 Ki = 4211 nM T76685 CM7DG0 127032456 IC50 > 10000 nM T76685 CBE3R6 127032540 Ki > 10000 nM T76685 C7L8BN 127032985 Ki = 1519 nM T76685 CA7HV0 127032986 Ki = 1172 nM T76685 C3YG8K 127033294 Ki > 10000 nM T76685 CUNJ13 127033295 Ki > 10000 nM T76685 C6JM5H 127033296 Ki > 10000 nM T76685 CSGK03 127033297 Ki > 10000 nM T76685 CZ73AN 127033298 Ki > 10000 nM T76685 CL47YF 127033299 Ki > 10000 nM T76685 C6XWZ5 127033300 Ki > 10000 nM T76685 CDFJ81 127033483 Ki > 40000 nM T76685 C2L0UO 127033585 Ki > 10000 nM T76685 C5WK8C 127033586 Ki > 10000 nM T76685 CXG07N 127033786 Ki > 40000 nM T76685 C8N0RD 127033787 Ki > 40000 nM T76685 CB9OZ6 127034064 Ki > 40000 nM T76685 C9D8NR 127034065 Ki > 40000 nM T76685 C30BCV 127034066 Ki > 40000 nM T76685 CK57OG 127034067 Ki > 40000 nM T76685 C4K9RW 127034068 Ki > 40000 nM T76685 CEH0S2 127034069 Ki > 40000 nM T76685 CD3K1V 127034070 Ki > 40000 nM T76685 CSK5Y7 127034071 Ki > 40000 nM T76685 C36TFY 127034072 Ki > 40000 nM T76685 C6GPQ0 127034073 Ki > 40000 nM T76685 C0KBT1 127034080 Ki > 40000 nM T76685 CQ9N4O 127034141 Ki = 4718 nM T76685 COA3U0 127034142 Ki = 5216 nM T76685 CST04W 127034143 Ki = 5849 nM T76685 CD4VN6 127034337 Ki > 10000 nM T76685 C56NPM 127034412 Ki = 3723 nM T76685 CE7U2X 127034413 Ki > 10000 nM T76685 C75HWE 127034414 Ki = 6352 nM T76685 CE51CW 127034415 Ki > 10000 nM T76685 C7LXG3 127045805 Ki >= 10000 nM T76685 CX40GI 127045919 Ki = 1557 nM T76685 CQ56AZ 127045920 Ki = 2502 nM T76685 C6AC8U 127046131 Ki = 380 nM T76685 CQ0FN3 127046132 Ki = 1070 nM T76685 C4QH0N 127046416 Ki = 2831 nM T76685 C5XD4U 127046684 Ki = 6111 nM T76685 C2BP4Q 127046685 Ki = 2523 nM T76685 C9PW8O 127046686 Ki = 904.5 nM T76685 CCU7A4 127046687 Ki = 826 nM T76685 C9DFA6 127047182 EC50 = 340 nM T76685 C28FLN 127047317 EC50 = 330 nM T76685 CU2ST0 127047318 EC50 = 270 nM T76685 C6TMB2 127047319 EC50 = 40 nM T76685 COLP16 127047329 Ki = 615 nM T76685 CGV6Y5 127047410 Ki = 1859 nM T76685 CY80XQ 127047411 Ki = 549 nM T76685 CB80KL 127047458 EC50 = 19 nM T76685 C1D7PX 127047462 EC50 = 310 nM T76685 C0RE8Z 127047592 EC50 = 9.1 nM T76685 C71MFW 127047640 EC50 = 200 nM T76685 C6P4OZ 127047641 EC50 = 4.4 nM T76685 CO0WB4 129257195 Ki > 10000 nM T76685 CL2A1B 129781980 Ki > 10000 nM T76685 C0ZYK8 130339702 Ki = 982 nM T76685 C50IHF 130339703 Ki = 1614 nM T76685 C8D3MY 130366796 Ki > 10000 nM T76685 CJHT67 132510986 Ki > 40000 nM T76685 CB1D8Q 132578438 Ki = 7000 nM T76685 C50HGD 132578440 Ki = 5700 nM T76685 C2AKW3 132585222 EC50 > 10000 nM T76685 CNSG54 132585223 EC50 > 10000 nM T76685 CDK60Q 134130813 Ki = 600 nM T76685 CDP7U0 134131733 Ki = 5100 nM T76685 C1Q9XZ 134131985 Ki > 10000 nM T76685 CF64DG 134132091 EC50 = 32 nM T76685 CLR9C6 134132855 Ki > 10000 nM T76685 C7B4JU 134133334 Ki = 3736.7 nM T76685 CWG8P2 134133524 Ki > 10000 nM T76685 CTI0Y2 134133618 Ki > 10000 nM T76685 CFTS48 134134129 EC50 = 8 nM T76685 CV8SR9 134134298 Ki > 10000 nM T76685 C7IEV8 134135104 EC50 = 24 nM T76685 C4ILM0 134135334 Ki > 10000 nM T76685 C7BQ5W 134135465 EC50 = 30 nM T76685 C5WFH6 134135522 EC50 = 7 nM T76685 COI6K4 134135649 Ki > 10000 nM T76685 CK0RA6 134135962 Ki = 4571.51 nM T76685 C3K9NQ 134136117 EC50 = 9 nM T76685 C4NBF7 134136193 EC50 = 5 nM T76685 C1ZW2U 134136510 Ki > 10000 nM T76685 C5JQ6R 134136907 EC50 = 12 nM T76685 C9J5KY 134137187 Ki > 10000 nM T76685 CUG02L 134137271 Ki > 10000 nM T76685 C32UGQ 134137479 Ki = 5926.7 nM T76685 CY2EK1 134137727 Ki > 10000 nM T76685 C3Y6FA 134138389 EC50 = 15 nM T76685 C0OHC7 134138469 EC50 = 7 nM T76685 C3J6GU 134138518 EC50 = 20 nM T76685 CW1KO0 134138598 Ki > 10000 nM T76685 CIM01Y 134138796 EC50 = 56 nM T76685 C7T2EY 134138952 EC50 = 28 nM T76685 CTZ5Q6 134139255 EC50 = 8 nM T76685 CGTZ26 134139273 EC50 = 18 nM T76685 C1NJ9C 134139421 Ki = 5900 nM T76685 CJ1FG3 134139799 Ki = 281.06 nM T76685 C4Z0KB 134140018 Ki > 10000 nM T76685 CDB9F4 134140655 EC50 = 28 nM T76685 C2QGM7 134140841 EC50 = 35 nM T76685 C1HD0Q 134140959 EC50 = 13 nM T76685 C6GJB1 134141428 Ki > 10000 nM T76685 CTZ4H5 134141506 Ki > 10000 nM T76685 C95QFU 134141929 EC50 = 6 nM T76685 CZ3H1I 134142321 Ki = 5100 nM T76685 CC4H7W 134142473 Ki > 10000 nM T76685 CITW76 134142657 EC50 = 4 nM T76685 CW4N6H 134142675 EC50 = 17 nM T76685 C5Y9UW 134142847 Ki = 5800 nM T76685 CGN42L 134143149 EC50 = 6 nM T76685 C2M9IN 134143205 EC50 = 18 nM T76685 CNT6D2 134143262 Ki = 700 nM T76685 CVT6D2 134144382 Ki > 10000 nM T76685 CNF1C8 134144706 Ki = 633.03 nM T76685 CL8T0G 134145050 EC50 = 37 nM T76685 CN7TR5 134145283 EC50 = 8 nM T76685 C4S2FX 134146248 Ki = 500 nM T76685 C3E4RW 134146777 EC50 = 6 nM T76685 CP82DL 134146936 EC50 = 11 nM T76685 C84IHR 134148177 Ki > 10000 nM T76685 CERX86 134148188 EC50 = 4 nM T76685 CUV40N 134148570 Ki > 10000 nM T76685 C89YTJ 134149018 Ki > 10000 nM T76685 CR64GQ 134149040 Ki > 10000 nM T76685 C07FSW 134149771 Ki = 2900 nM T76685 CH9DW2 134149775 EC50 = 8 nM T76685 CBF56O 134149796 EC50 = 6 nM T76685 C1W4ID 134149884 EC50 = 2 nM T76685 C97HGO 134150139 Ki > 10000 nM T76685 C5IXY8 134150287 Ki = 2621.82 nM T76685 C5YG9D 134150307 EC50 = 22 nM T76685 C7TJY0 134150441 Ki = 317.03 nM T76685 CU63GK 134151463 EC50 = 37 nM T76685 CPZR93 134152278 EC50 = 17 nM T76685 CHA9B0 134152389 EC50 = 12 nM T76685 C8NGJ4 134152497 EC50 = 30 nM T76685 CG6M0R 134152684 EC50 = 7 nM T76685 CED06W 134154057 Ki > 10000 nM T76685 CJX45N 134154719 EC50 = 34 nM T76685 CC5TU4 134154932 EC50 = 28 nM T76685 CZOY08 134155237 EC50 = 4 nM T76685 C0MVG7 134155406 Ki = 1196.7 nM T76685 CJ1BA3 134155808 EC50 = 11 nM T76685 CML28S 134155966 Ki = 4600 nM T76685 C8QIC2 134156159 EC50 = 15 nM T76685 C0M2GZ 134156537 Ki > 10000 nM T76685 C6KS0N 134156578 Ki = 4900 nM T76685 C92VRD 134156729 Ki = 505.03 nM T76685 CEW50T 134156883 EC50 = 35 nM T76685 CYCE87 134157291 Ki > 10000 nM T76685 C0JL7I 134157399 EC50 = 22 nM T76685 CYS3B9 134157891 EC50 = 127 nM T76685 CNX5J2 134157932 Ki = 518.2 nM T76685 CNDI28 135156076 Ki = 2 nM T76685 CK8T9E 135156097 Ki = 12 nM T76685 CX2SZ4 135156106 Ki = 7 nM T76685 C1W9FV 135156138 Ki = 5 nM T76685 C7UJ0A 135156140 Ki = 4 nM T76685 CIS28F 135156142 Ki = 2 nM T76685 C7B0UK 135156143 Ki = 24 nM T76685 CN83XY 135156151 Ki = 12 nM T76685 CWEU47 135156153 Ki = 2 nM T76685 COC48A 135156160 Ki = 22 nM T76685 CGBP75 135156161 Ki = 8 nM T76685 CYE13V 135156182 Ki = 420 nM T76685 C0BLS7 135156185 Ki = 8 nM T76685 CF29ML 135156190 Ki = 0.38 nM T76685 CWU6L2 135156193 Ki = 1.4 nM T76685 CS9RP5 135156203 Ki = 8 nM T76685 CLS4A8 135156215 Ki = 8 nM T76685 CUI9X6 135156216 Ki = 14 nM T76685 CED38C 135156219 Ki = 24 nM T76685 C8BZ2J 135156223 Ki = 1.2 nM T76685 C0UO9X 135156228 Ki = 22 nM T76685 C4K1NW 135156229 Ki = 3 nM T76685 CXV38J 135156232 Ki = 5 nM T76685 CM4LS9 135156237 Ki = 25 nM T76685 C5U9ZM 135156239 Ki = 3 nM T76685 CA82SP 135156240 Ki = 3 nM T76685 CY8D4L 135156241 Ki = 0.6 nM T76685 CJ85SW 135156242 Ki = 2 nM T76685 C1GY2T 135156251 Ki = 22 nM T76685 CINV95 135156278 Ki = 4 nM T76685 C4C8FY 135156279 Ki = 4 nM T76685 CX8JS3 135156281 Ki = 6 nM T76685 C3AYS7 135156282 Ki = 6 nM T76685 C4Y3XH 135156284 Ki = 18 nM T76685 CQW0X9 135156285 Ki = 6 nM T76685 COW34N 135156292 Ki = 17 nM T76685 CR4A9I 135156296 Ki = 5 nM T76685 CK2C8T 135156317 Ki = 120 nM T76685 C5VA0M 135156319 Ki = 2 nM T76685 C0GE5U 135156322 Ki = 51 nM T76685 C1NX8O 135156329 Ki = 19 nM T76685 C5YP0R 135156335 Ki = 1 nM T76685 CSX16V 135156341 Ki = 2 nM T76685 CUE5F7 135156347 Ki = 5 nM T76685 CXT1L3 135156354 Ki = 5 nM T76685 CL6P8W 135156382 Ki = 3.3 nM T76685 CNW3I9 135156391 Ki = 2 nM T76685 CR29YT 135156426 Ki = 2 nM T76685 CN2RT9 135156435 Ki = 3 nM T76685 CDY28G 135156437 Ki = 26 nM T76685 C6L3MW 135156439 Ki = 2 nM T76685 CFU36D 135156440 Ki = 1 nM T76685 CQ7O9J 135156442 Ki = 5 nM T76685 C2HPY7 135156445 Ki = 4 nM T76685 CR1Z4C 135156452 Ki = 3 nM T76685 C7L6QM 135156454 Ki = 10 nM T76685 CNMF20 135156469 Ki = 7 nM T76685 CBSC28 135156470 Ki = 2 nM T76685 C7YIQ0 135156473 Ki = 24 nM T76685 CYML32 135156477 Ki = 3 nM T76685 C2WB5Y 135156479 Ki = 730 nM T76685 C25ENA 135156501 Ki = 1.7 nM T76685 C3NQ7M 135156503 Ki = 6 nM T76685 CBV81U 135156509 Ki = 0.9 nM T76685 CVW76H 135156513 Ki = 2 nM T76685 CJM59S 135164381 Ki = 5 nM T76685 C80TDY 135164613 Ki = 42 nM T76685 C92DIW 135165004 Ki = 780 nM T76685 C19PYU 135165007 Ki = 5 nM T76685 CP4EC6 135376107 IC50 = 1570 nM T76685 CI7C2K 135376115 IC50 = 169 nM T76685 C5AO6Y 135376117 IC50 = 95 nM T76685 CZX40L 135376124 IC50 = 164 nM T76685 C9L7GV 135376125 IC50 = 133 nM T76685 CZG91R 135376128 IC50 = 334 nM T76685 C7USA2 135376152 IC50 = 195 nM T76685 CLB40M 135376155 IC50 = 81 nM T76685 C3NJ8T 135376158 IC50 = 22 nM T76685 CP5BO2 135376159 IC50 = 47 nM T76685 CIM6W5 135376334 IC50 = 132 nM T76685 C3ROX7 135376339 IC50 = 30 nM T76685 C3J9LY 135376383 IC50 = 1260 nM T76685 C0YQS9 135376385 IC50 = 1310 nM T76685 CY9M3O 135376387 IC50 = 290 nM T76685 CA3S6K 135376388 IC50 = 27 nM T76685 CON12D 135376389 IC50 = 18 nM T76685 CK4S8X 135376391 IC50 = 40 nM T76685 CZ9C4I 135376399 IC50 = 178 nM T76685 C3XV6H 135376400 IC50 = 516 nM T76685 CH1B8A 135376403 IC50 = 591 nM T76685 C2SY0Q 135376412 IC50 = 231 nM T76685 CH1P0V 135376438 IC50 = 70 nM T76685 CHC95M 135376458 IC50 = 840 nM T76685 CBFG01 135376463 IC50 = 440 nM T76685 CB72ZS 135376465 IC50 = 338 nM T76685 C69SIB 135376559 IC50 = 460 nM T76685 CDF8R7 135376575 IC50 = 32 nM T76685 CJAS26 135376577 IC50 = 134 nM T76685 CZ10DT 135376603 IC50 = 190 nM T76685 CJ40GC 135376608 IC50 = 35 nM T76685 CC4DN5 135376614 IC50 = 244 nM T76685 C54DNJ 135376621 IC50 = 1340 nM T76685 C98IOH 135376632 IC50 = 42 nM T76685 C31YBD 135376656 IC50 = 74 nM T76685 CD3V1F 135376751 IC50 = 23 nM T76685 C3MTP9 135446388 IC50 = 251.19 nM T76685 C7L4DP 135547119 IC50 = 125 nM T76685 CTA68K 135881483 EC50 = 937.1 nM T76685 C0R5SW 135881484 EC50 = 852 nM T76685 CSB01I 135881485 EC50 = 62.3 nM T76685 CRQ1H4 135922724 IC50 = 200 nM T76685 C8UG5X 135922725 IC50 = 400 nM T76685 CI86RJ 135923581 IC50 = 130 nM T76685 C04MQH 135923694 IC50 = 7.4 nM T76685 C8DOW1 135923695 IC50 = 6 nM T76685 CUQC19 135923696 IC50 = 59 nM T76685 CO3SU7 135924633 EC50 > 10000 nM T76685 C28CMN 135924634 EC50 = 263 nM T76685 CF17PG 135924635 EC50 > 10000 nM T76685 C1Y6IV 135924636 EC50 = 61.2 nM T76685 CQFV38 135924637 EC50 > 10000 nM T76685 CWH7R6 135924638 EC50 > 10000 nM T76685 CH5MI8 135924639 EC50 > 10000 nM T76685 CO2FL0 135924640 EC50 > 10000 nM T76685 C0OP6U 135924641 EC50 > 10000 nM T76685 C2XBO9 135924642 EC50 > 10000 nM T76685 CIGQ76 135924643 EC50 > 10000 nM T76685 CH37QR 135924644 EC50 > 10000 nM T76685 C8F4SQ 135924645 EC50 > 10000 nM T76685 CI4SU6 135924646 EC50 > 10000 nM T76685 CDL89Z 135924647 EC50 > 10000 nM T76685 C04MZE 135930698 EC50 = 459 nM T76685 C9ROE1 135936176 Ki = 28.5 nM T76685 CE26DH 135936177 Ki = 14.2 nM T76685 C0WB3A 135936178 Ki = 4.5 nM T76685 CXH73Y 135936179 Ki = 18.6 nM T76685 CCOB67 135936180 Ki = 514 nM T76685 CD3K1W 135936181 Ki = 5.2 nM T76685 CSRK39 135995913 EC50 > 10000 nM T76685 C8S1ME 135995914 EC50 > 10000 nM T76685 CI7Z5E 135995915 EC50 > 10000 nM T76685 C2RG1O 135995916 EC50 > 10000 nM T76685 CVZ6G2 135995917 EC50 > 10000 nM T76685 C0RH1T 135995918 EC50 > 10000 nM T76685 C31RKJ 135995919 EC50 > 10000 nM T76685 C0DQ2F 135995920 EC50 > 10000 nM T76685 C1APX3 135995921 EC50 > 10000 nM T76685 CTG9L5 135995922 EC50 > 10000 nM T76685 C5O9AI 135995923 EC50 > 10000 nM T76685 CNHL53 135995924 EC50 > 10000 nM T76685 C36XJL 135995925 EC50 > 10000 nM T76685 CG7C6Z 135995926 EC50 > 10000 nM T76685 COR21T 135995927 EC50 > 10000 nM T76685 CXC32Y 135995928 EC50 > 10000 nM T76685 C39DSU 135995929 EC50 > 10000 nM T76685 C3TWF4 135995930 EC50 > 10000 nM T76685 CA6RF7 135995931 EC50 > 10000 nM T76685 C0LJQ3 135995932 EC50 > 10000 nM T76685 C74RUI 135995933 EC50 > 10000 nM T76685 CXF8I9 135995934 EC50 > 10000 nM T76685 C0W6AO 135995935 EC50 > 10000 nM T76685 C86KWU 135995936 EC50 > 10000 nM T76685 C5TOD3 135995937 EC50 > 10000 nM T76685 CDL8C1 135995938 EC50 > 10000 nM T76685 C5TF8G 135995939 EC50 > 10000 nM T76685 C2E5KG 135995940 EC50 > 10000 nM T76685 CDQ54M 135995941 EC50 > 10000 nM T76685 CNC8O4 135995942 EC50 > 10000 nM T76685 CA8QI4 135995943 IC50 > 10000 nM T76685 C30QJD 135995944 IC50 > 10000 nM T76685 CT3DY8 135995945 IC50 > 10000 nM T76685 CTX8Y4 135995946 IC50 > 10000 nM T76685 CG8H3C 135995947 IC50 > 10000 nM T76685 CJ4W5Y 135995948 IC50 > 10000 nM T76685 C4AQC1 135995949 IC50 > 10000 nM T76685 C9JBO5 135995950 IC50 > 10000 nM T76685 C42UVC 135995951 IC50 > 10000 nM T76685 CO8PT2 136045810 EC50 = 1238.8 nM T76685 CQFZ04 136059727 IC50 = 2500 nM T76685 CP0VN6 136141590 EC50 <= 100 nM T76685 CL8MD3 136180708 Ki = 5.2 nM T76685 C2A3KM 136180709 Ki = 9.5 nM T76685 CW0OS1 136266294 IC50 > 10000 nM T76685 C86HUN 136266296 IC50 > 10000 nM T76685 CV9J6O 136266306 IC50 > 10000 nM T76685 C8EIW4 136266307 IC50 > 10000 nM T76685 CP17HJ 136266308 IC50 > 10000 nM T76685 C1M7XU 136266314 IC50 > 10000 nM T76685 CGE38A 136266318 IC50 > 10000 nM T76685 C7AU4T 136266319 EC50 > 10000 nM T76685 C5EB1A 136266320 EC50 > 10000 nM T76685 CNAG68 136266324 EC50 > 10000 nM T76685 CD75IA 136266326 IC50 > 10000 nM T76685 C7SGJ1 136266328 IC50 > 10000 nM T76685 CNT63W 137062188 EC50 = 2020 nM T76685 CD7B2E 137062189 EC50 > 10000 nM T76685 CIP3Z7 137062190 EC50 > 10000 nM T76685 C3A0PC 137062191 EC50 > 10000 nM T76685 C43HNY 137062192 EC50 = 557 nM T76685 C40YWC 137062193 EC50 > 10000 nM T76685 C9G4KR 137062194 EC50 > 10000 nM T76685 CYBZ12 137169067 EC50 = 63.1 nM T76685 CPW0D2 137346241 EC50 = 2100 nM T76685 C61JRN 137346243 EC50 = 180 nM T76685 CE9HS4 137346244 EC50 = 151.36 nM T76685 C45CDW 137631524 EC50 = 13000 nM T76685 C03ECM 137632290 EC50 = 6700 nM T76685 C92XMB 137632971 EC50 > 10000 nM T76685 CH0B6U 137634141 EC50 > 10000 nM T76685 CEX02D 137634149 EC50 > 10000 nM T76685 CY5UW7 137634172 Ki > 4000 nM T76685 CRA1X6 137634457 Ki > 4000 nM T76685 C3CT4W 137635042 EC50 > 10000 nM T76685 CV97TL 137635223 EC50 > 10000 nM T76685 CF13WZ 137635764 EC50 > 10000 nM T76685 C1DUY6 137636294 IC50 = 141 nM T76685 CI5B1C 137636709 EC50 > 10000 nM T76685 CR7N8A 137637773 EC50 > 10000 nM T76685 C4IC9D 137637998 EC50 > 10000 nM T76685 CDZW38 137638255 Ki = 245 nM T76685 CG16DR 137638994 Ki > 1000 nM T76685 C5A7DC 137639252 EC50 > 10000 nM T76685 C8XHT3 137639360 Ki > 4000 nM T76685 C5HV6S 137639623 EC50 > 10000 nM T76685 C2GEU5 137639906 Ki > 1000 nM T76685 CU8TJ5 137640021 Ki = 2.512 nM T76685 CME1D4 137640026 EC50 > 10000 nM T76685 CCY7B8 137640363 Ki = 1000 nM T76685 C1M7NV 137640777 EC50 = 3300 nM T76685 C4TUW2 137640869 EC50 > 10000 nM T76685 CUE37K 137641100 EC50 > 10000 nM T76685 C98FBN 137642085 Ki > 4000 nM T76685 CEYG80 137642209 Ki > 1000 nM T76685 CH80BJ 137643152 EC50 > 10000 nM T76685 CCBH92 137643269 EC50 > 10000 nM T76685 CWA3I4 137643432 EC50 > 10000 nM T76685 CI6NL3 137643518 Ki > 4000 nM T76685 CXER43 137644281 EC50 > 10000 nM T76685 CLN0W5 137644328 Ki = 25 nM T76685 CR25ML 137644618 EC50 = 630 nM T76685 CAN3G2 137645158 Ki > 4000 nM T76685 CNGB09 137645429 EC50 > 10000 nM T76685 CP9LT8 137647595 EC50 > 10000 nM T76685 CETC84 137647970 EC50 > 10000 nM T76685 C68HNE 137648160 EC50 > 10000 nM T76685 C5M2VE 137648805 Ki = 1100 nM T76685 C26JNU 137649145 EC50 > 10000 nM T76685 CVF9U7 137649354 EC50 = 84 nM T76685 C9OYR4 137650162 EC50 > 10000 nM T76685 C4QFY0 137650412 EC50 > 10000 nM T76685 C2AS9T 137650812 EC50 = 4100 nM T76685 CK7RD3 137650977 Ki = 467 nM T76685 CWZ92Q 137651267 IC50 > 10000 nM T76685 C3WI7F 137652938 EC50 > 10000 nM T76685 CIJW29 137653436 EC50 > 10000 nM T76685 CS13JP 137654029 Ki = 115 nM T76685 CCJ74L 137654157 EC50 > 10000 nM T76685 CI18ZR 137654462 EC50 > 10000 nM T76685 CPS17B 137654744 EC50 > 10000 nM T76685 C02YDQ 137655423 Ki > 4000 nM T76685 C10OJC 137655779 EC50 > 10000 nM T76685 C4HA0W 137655793 Ki > 4000 nM T76685 C3P0YS 137655815 EC50 > 10000 nM T76685 CE86PO 137657290 EC50 = 22 nM T76685 C6GBO0 137657351 EC50 > 10000 nM T76685 CQC6G7 137658542 IC50 = 15848.93 nM T76685 C5LC2S 137658778 Ki = 365 nM T76685 CG5BW8 137658946 Ki = 33 nM T76685 CO1SG5 137659148 EC50 > 10000 nM T76685 CK0AC9 137660701 Ki = 1000 nM T76685 CY93TX 137661282 EC50 > 10000 nM T76685 CP5QB4 137662088 EC50 > 10000 nM T76685 CB8IM1 138319671 IC50 > 10000 nM T76685 C4SY8V 138491556 EC50 = 0.03 nM T76685 C82LVN 138491578 EC50 = 0.07 nM T76685 CZQ61R 138491579 EC50 = 0.19 nM T76685 CK6HN2 140685644 Ki = 436 nM T76685 CA07WZ 141463725 EC50 > 10000 nM T76685 C2XU4C 141463726 EC50 = 2605 nM T76685 CPZ62D 141463727 EC50 > 10000 nM T76685 CYU0K3 141463728 EC50 > 10000 nM T76685 CINT06 141463729 EC50 > 10000 nM T76685 C2FMK0 141463730 EC50 > 10000 nM T76685 C7I8XT 141463734 EC50 > 10000 nM T76685 C93LEZ 141463736 EC50 > 10000 nM T76685 CHDV64 141463737 EC50 > 10000 nM T76685 CTGM15 141463743 EC50 > 10000 nM T76685 CJA91I 141463744 EC50 > 10000 nM T76685 C1MSD2 141463745 EC50 > 10000 nM T76685 CXY8V2 141463746 EC50 > 10000 nM T76685 CET5X6 141463751 EC50 > 10000 nM T76685 CYI8H5 141463752 EC50 > 10000 nM T76685 C4F7KJ 141463753 EC50 > 10000 nM T76685 CGL2O4 141463754 EC50 > 10000 nM T76685 C8GO7V 141463760 EC50 > 10000 nM T76685 CKXG28 141463761 EC50 > 10000 nM T76685 CZ02KM 141463762 EC50 > 10000 nM T76685 CJY41G 141463764 EC50 > 10000 nM T76685 C2KJ9N 141463766 EC50 > 10000 nM T76685 C4HF2M 141463767 EC50 > 10000 nM T76685 C7AO1T 141463769 EC50 > 10000 nM T76685 CZL4T6 141463770 EC50 > 10000 nM T76685 C39QOI 141463775 EC50 > 10000 nM T76685 C61RIQ 141463776 EC50 = 10000 nM T76685 C6WQI5 141463778 EC50 = 6047 nM T76685 C1OY9J 141463781 EC50 > 10000 nM T76685 C1F0BP 145949413 Ki > 10000 nM T76685 CBC13V 145949551 Ki > 10000 nM T76685 C5XM3H 145949852 Ki > 10000 nM T76685 CSI2U8 145949897 Ki > 1000 nM T76685 C1PH6E 145949978 Ki > 1000 nM T76685 CXRO20 145950071 Ki > 10000 nM T76685 CY60SW 145951064 Ki > 10000 nM T76685 CCKN03 145951123 Ki > 10000 nM T76685 CSM7J0 145951205 Ki > 10000 nM T76685 CSG0W9 145951227 Ki > 10000 nM T76685 C8EV4M 145951290 Ki > 1000 nM T76685 C4LX7H 145951404 Ki > 10000 nM T76685 C4IX1W 145951504 Ki = 30.7 nM T76685 C24POL 145951821 Ki > 1000 nM T76685 CS09YQ 145951898 Ki = 293 nM T76685 C06VUY 145951905 Ki = 113 nM T76685 C6NXD2 145952218 Ki > 1000 nM T76685 C3G5TZ 145952824 Ki > 10000 nM T76685 CS10GA 145953541 Ki > 10000 nM T76685 CDE1H5 145953638 Ki > 1000 nM T76685 CV0S3L 145953742 Ki > 10000 nM T76685 CDI42H 145953879 Ki > 10000 nM T76685 CMZ2B1 145953904 Ki > 1000 nM T76685 CSHA03 145953939 IC50 = 14130 nM T76685 CZK20O 145954166 Ki > 1000 nM T76685 C6QX5T 145954189 Ki > 10000 nM T76685 CKO9B4 145954190 Ki > 10000 nM T76685 CF63TZ 145954337 IC50 = 100000 nM T76685 COMQ03 145954409 Ki = 1670 nM T76685 C7N1JT 145954513 IC50 > 10000 nM T76685 CN7K2W 145954743 Ki > 1000 nM T76685 C03WAH 145954816 Ki > 10000 nM T76685 CVL21U 145954925 Ki > 1000 nM T76685 CUE8Y2 145955444 Ki > 10000 nM T76685 C2KJ8F 145955689 Ki = 23.1 nM T76685 CX95DH 145955833 Ki > 10000 nM T76685 C46LCZ 145955918 Ki > 10000 nM T76685 CDG60N 145956233 EC50 > 10000 nM T76685 CG16ZX 145956544 Ki > 10000 nM T76685 CP0L8K 145956576 Ki > 10000 nM T76685 CA30EJ 145956612 Ki > 10000 nM T76685 CEX3U4 145956825 Ki = 131 nM T76685 CX20FR 145956970 IC50 > 100000 nM T76685 C16HBG 145956992 Ki > 1000 nM T76685 CX70KY 145957108 Ki > 10000 nM T76685 C1CAR4 145957287 Ki > 1000 nM T76685 CG6YU8 145957460 EC50 > 10000 nM T76685 CR8E3C 145957540 Ki > 1000 nM T76685 C4AUS9 145957967 EC50 = 0.43 nM T76685 CW3A0Y 145958034 Ki = 2210 nM T76685 CIK3B7 145958405 Ki > 10000 nM T76685 CC5B9Y 145958428 Ki > 10000 nM T76685 C1S8TU 145958458 IC50 = 17920 nM T76685 C3IH1U 145958480 Ki > 10000 nM T76685 COP8M1 145958551 Ki > 10000 nM T76685 CEQ9W7 145958588 Ki > 10000 nM T76685 CZ1N2I 145958910 Ki > 1000 nM T76685 CATQ56 145959099 IC50 > 100000 nM T76685 C5K9TY 145959141 Ki > 10000 nM T76685 CEUL02 145959311 EC50 > 10000 nM T76685 CDEK59 145959588 EC50 = 1.4 nM T76685 C25PYN 145959820 Ki > 1000 nM T76685 CLP94K 145960053 Ki > 1000 nM T76685 C25WFH 145960085 Ki > 10000 nM T76685 CQ3B6P 145960178 Ki > 10000 nM T76685 CVHI05 145961169 EC50 > 10000 nM T76685 CFV4A7 145962733 EC50 > 10000 nM T76685 CA5S6Z 145964684 Ki = 246.6 nM T76685 COB60Z 145964887 Ki = 3604 nM T76685 C5RH7P 145965270 Ki > 10000 nM T76685 C47YHA 145965727 Ki = 707.6 nM T76685 C09BZG 145965919 IC50 = 1900 nM T76685 C5WN1R 145966442 Ki = 1248 nM T76685 CKQU13 145967105 Ki = 1462 nM T76685 CU1O5Y 145968444 Ki = 73.2 nM T76685 C0ST1H 145968723 Ki = 44.6 nM T76685 C96LYC 145968771 Ki = 4 nM T76685 CNK2J9 145969213 Ki = 7 nM T76685 CX8I0M 145970908 Ki = 1.1 nM T76685 C5T2WE 145971274 Ki > 10000 nM T76685 C46CJZ 145971303 Ki = 724.2 nM T76685 C6XAW4 145971463 Ki > 10000 nM T76685 CU3V6E 145971521 Ki > 1000 nM T76685 CDN40B 145972411 Ki = 11.7 nM T76685 CVI92K 145972432 Ki > 1000 nM T76685 CHUV20 145972574 Ki = 800.4 nM T76685 CVL6X0 145972916 IC50 > 100000 nM T76685 C41SIK 145973984 Ki = 1286 nM T76685 C4G8WI 145974549 Ki > 10000 nM T76685 CR2I5X 145974580 IC50 > 10000 nM T76685 C09DRX 145974911 Ki > 40000 nM T76685 COQP62 145975266 Ki = 1193 nM T76685 CP8A5L 145975353 Ki = 856.5 nM T76685 CK8S6G 145975678 Ki = 75.5 nM T76685 C8OER4 145976515 Ki > 10000 nM T76685 CWKV12 145976995 Ki > 40000 nM T76685 CVS75Z 145977686 Ki = 608.8 nM T76685 CKT7O8 145977995 IC50 = 9600 nM T76685 CY34IF 145978111 IC50 = 180 nM T76685 C8PSE7 145979528 EC50 = 632.5 nM T76685 C8O1FW 145979865 Ki > 10000 nM T76685 C2GBD6 145980256 EC50 = 260 nM T76685 CR7VZ6 145980710 EC50 > 10000 nM T76685 C4I1NP 145981357 Ki > 10000 nM T76685 CV0Z9N 145982058 Ki > 10000 nM T76685 C65SRO 145982136 EC50 = 4900 nM T76685 C20OQS 145982249 EC50 = 113 nM T76685 C3EAH9 145982250 Ki = 193 nM T76685 CGD26R 145982389 EC50 = 77 nM T76685 CLP8R3 145982513 Ki = 11 nM T76685 CZ8Q6U 145982659 Ki = 3 nM T76685 C8OMN3 145983082 Ki = 13 nM T76685 CP95QD 145983220 Ki = 3 nM T76685 C29YPO 145983245 Ki = 43 nM T76685 CP0AW6 145983324 Ki = 3 nM T76685 CZ0O2J 145983660 Ki > 10000 nM T76685 CZ64LM 145983702 Ki > 10000 nM T76685 C2O3KS 145984100 Ki = 2 nM T76685 CM2U6K 145984485 Ki = 250 nM T76685 C8NI7A 145984522 Ki = 1.7 nM T76685 CK3PA7 145984774 Ki = 1.4 nM T76685 CFL94B 145984952 Ki = 1.2 nM T76685 CWV57R 145985098 Ki = 2 nM T76685 CQ96YL 145985429 Ki = 3 nM T76685 CXI7F5 145985700 Ki = 21 nM T76685 CF4P2L 145985979 Ki = 0.4 nM T76685 C6N8ER 145986153 Ki = 8 nM T76685 CC1F5K 145986420 Ki = 286 nM T76685 C53WHL 145986477 EC50 = 322 nM T76685 CS0N5V 145987144 Ki = 48 nM T76685 CHOY46 145987281 Ki = 12 nM T76685 C6TS3J 145987421 Ki > 10000 nM T76685 C7EX9O 145987549 EC50 = 126 nM T76685 CV1IH0 145988362 IC50 = 4100 nM T76685 C3X0BU 145988575 EC50 = 66 nM T76685 C5WF0E 145988921 Ki > 10000 nM T76685 C08SWB 145988974 Ki = 642 nM T76685 CDK37M 145988985 Ki = 823.8 nM T76685 CNP5G9 145989291 Ki = 919 nM T76685 CK74GP 145989580 Ki > 10000 nM T76685 CEK4P6 145989716 Ki = 3 nM T76685 C0B7HW 145990576 EC50 = 62.9 nM T76685 C6UC1D 145990629 EC50 = 1150 nM T76685 CK8BM3 145990869 Ki = 538 nM T76685 CL15JC 145990912 Ki = 4527 nM T76685 C0ULZ5 145990999 IC50 = 2600 nM T76685 C4MPJ3 145991020 Ki > 10000 nM T76685 CGR85Q 145991514 EC50 > 10000 nM T76685 CT4GP2 145991901 Ki = 2850 nM T76685 CSWZ43 145992799 EC50 = 5 nM T76685 CZ9PB3 145993004 Ki = 1583 nM T76685 CCH5P9 145993268 Ki = 512 nM T76685 CPBZ37 145993775 Ki = 504.6 nM T76685 CA6BY0 145993873 Ki = 1400 nM T76685 CXHY67 145993892 Ki = 3918 nM T76685 CK6F7I 145994018 Ki > 10000 nM T76685 CYXP50 146257099 Ki = 5 nM T76685 CR2Q4T 146257107 Ki = 2.4 nM T76685 C93MHJ 146257111 Ki = 47 nM T76685 C6REF2 146257116 Ki = 6 nM T76685 C1KX0T 147088776 EC50 = 5528 nM T76685 CDO41B 153544782 IC50 = 4 nM T76685 C6YKS5 153544784 IC50 = 3 nM T76685 CBZ1D9 155436492 IC50 = 39 nM T76685 CX3IL7 155436493 IC50 = 5020 nM T76685 CY2JF6 155436497 IC50 = 61 nM T76685 CM8F5W 155436500 IC50 = 156 nM T76685 CXIM05 155436502 IC50 = 92 nM T76685 C3MW1Y 155436503 IC50 = 233 nM T76685 C2NYA7 155436506 IC50 = 111 nM T76685 CO76PL 155436509 IC50 = 79 nM T76685 C5B8RA 155436510 IC50 = 1270 nM T76685 C2X1AI 155436512 IC50 = 31 nM T76685 CB97LM 155436516 IC50 = 501 nM T76685 C4NBG5 155436589 IC50 = 21 nM T76685 CA5PI0 155436641 IC50 = 48 nM T76685 CG3PD5 155436644 IC50 = 40 nM T76685 CJDI76 155436645 IC50 = 37 nM T76685 CJPO29 155436648 IC50 = 3530 nM T76685 C9WE0U 155436651 IC50 = 58 nM T76685 CD05BE 155436652 IC50 = 2530 nM T76685 CFQ4O8 155436703 IC50 = 43 nM T76685 CV7M3Q 155436704 IC50 = 108 nM T76685 C2IKU4 155436706 IC50 = 40 nM T76685 C1T7KE 155436714 IC50 = 22 nM T76685 CG5M0C 155436719 IC50 = 60 nM T76685 CYB9R4 155436729 IC50 = 3880 nM T76685 C3ZT6B 155436731 IC50 = 292 nM T76685 CF9QM6 155436767 IC50 = 107 nM T76685 CCM50S 155491029 EC50 = 14 nM T76685 C98IPE 155510384 IC50 > 1000 nM T76685 C0AZ2W 155510575 IC50 > 10000 nM T76685 CJ56ZF 155511536 Ki = 671.3 nM T76685 C5BFO4 155511580 Ki = 19 nM T76685 C4GZ8M 155512603 Ki > 10000 nM T76685 CQ68IY 155512632 Ki > 10000 nM T76685 CY42GK 155512680 Ki = 0.1 nM T76685 CP69DA 155512716 Ki > 10000 nM T76685 C5YR0F 155512740 Ki = 2324 nM T76685 C6DGX2 155512779 IC50 > 1000 nM T76685 CBK10F 155513149 Ki = 9 nM T76685 C5LS3N 155513448 EC50 > 10000 nM T76685 C5HR6N 155513497 EC50 = 1100 nM T76685 C8W7IC 155513659 Ki = 657 nM T76685 C21PQJ 155514226 EC50 > 100000 nM T76685 C71HXW 155514525 Ki = 4414 nM T76685 CXPO26 155514667 Ki = 81 nM T76685 C19CSO 155514785 EC50 = 113 nM T76685 CC60EO 155514861 Ki = 1.6 nM T76685 C7HN4W 155514938 Ki = 1324 nM T76685 C5AJ0D 155515105 Ki = 2 nM T76685 CK2N9G 155515441 Ki = 1100 nM T76685 CRDT78 155515622 Ki = 19.1 nM T76685 CV3TS9 155515668 Ki = 450.4 nM T76685 C5Q7TM 155515733 EC50 = 56 nM T76685 C8WO0D 155515901 IC50 > 10000 nM T76685 C37OWC 155516090 Ki = 780 nM T76685 C7PNV4 155516299 Ki = 131 nM T76685 CQ7KF5 155516555 Ki = 2200 nM T76685 C5DPB7 155516636 Ki > 40000 nM T76685 CC0TY5 155516728 Ki = 1613 nM T76685 COAX01 155516832 Ki = 15 nM T76685 CGI38A 155516835 IC50 = 1220 nM T76685 CX7C2A 155517217 Ki = 260 nM T76685 CXCY52 155517496 Ki = 3 nM T76685 CDK74C 155517745 Ki > 10000 nM T76685 C8TS4W 155517909 IC50 > 1000 nM T76685 CCB70X 155518661 Ki = 3 nM T76685 C4GY3D 155519492 Ki > 10000 nM T76685 CTH10C 155519694 Ki = 2930 nM T76685 C38VFS 155519822 EC50 = 710 nM T76685 C0HSD3 155519911 IC50 > 10000 nM T76685 C7N4IS 155519912 Ki > 40000 nM T76685 CCG97Q 155519954 Ki = 9 nM T76685 CKMG08 155519959 EC50 = 29200 nM T76685 C0YW6N 155520181 Ki = 0.9 nM T76685 C2SV1D 155520325 Ki > 10000 nM T76685 C0YKO4 155520531 Ki = 45 nM T76685 CEN8W5 155520642 EC50 = 650 nM T76685 C6FQ5C 155520810 Ki = 3 nM T76685 CUL1B4 155521239 Ki = 1693 nM T76685 C6P2CJ 155521466 Ki = 1.2 nM T76685 CHUL10 155521781 EC50 = 130 nM T76685 CV0E2Y 155522138 Ki = 5040 nM T76685 C7NG1E 155522628 Ki = 2.6 nM T76685 CGO6N9 155523238 Ki = 106 nM T76685 C42TIR 155523370 Ki = 6 nM T76685 C2ES7G 155523649 Ki = 80 nM T76685 CV9U0X 155524379 EC50 = 158 nM T76685 C0O4YW 155525197 EC50 > 10000 nM T76685 CGP6I0 155525267 EC50 = 824 nM T76685 C5BCZ4 155525275 IC50 = 300 nM T76685 C3CS7M 155525734 IC50 = 40 nM T76685 CAP1Q4 155525954 Ki = 3770 nM T76685 C3NYA9 155526609 IC50 > 10000 nM T76685 C6RK9Y 155526850 Ki > 40000 nM T76685 C1XSG2 155526874 IC50 = 12 nM T76685 C63WYD 155527699 Ki > 10000 nM T76685 CFSY21 155527981 EC50 = 43 nM T76685 CN12US 155528165 Ki = 2110 nM T76685 C8IEW7 155528485 Ki > 10000 nM T76685 CN8V9G 155528513 Ki > 10000 nM T76685 C5NA1U 155528573 IC50 > 10000 nM T76685 C2WVB8 155529389 Ki = 0.26 nM T76685 CUZ7H8 155529444 Ki > 10000 nM T76685 CRS13Y 155529582 Ki = 58.89 nM T76685 C0JOP1 155529628 Ki > 10000 nM T76685 C19JGM 155530434 EC50 = 450 nM T76685 C7IMV5 155530567 IC50 > 10000 nM T76685 CS89CY 155531278 Ki = 22.4 nM T76685 C6Z9GK 155531741 IC50 > 10000 nM T76685 CBG1Z4 155531768 Ki = 4 nM T76685 C9GOV6 155531899 Ki = 0.8 nM T76685 CPI0E3 155531980 Ki > 40000 nM T76685 CVK1F0 155532408 EC50 = 2.2 nM T76685 CCF52B 155532449 IC50 > 1000 nM T76685 CFCE85 155532563 Ki > 10000 nM T76685 CAN9V6 155533000 Ki = 6 nM T76685 CGS63L 155533300 IC50 > 10000 nM T76685 CU5Q7F 155533412 Ki > 10000 nM T76685 C9NYQ7 155533629 EC50 = 230 nM T76685 C7OKT0 155533651 Ki = 0.2 nM T76685 CI3L5S 155534105 Ki = 6000 nM T76685 CLG6M7 155534607 Ki > 10000 nM T76685 C1J8PF 155534724 EC50 = 270 nM T76685 CF1J9O 155534934 Ki = 13 nM T76685 C50YMD 155535235 Ki > 10000 nM T76685 C1APZ8 155535329 Ki = 1660 nM T76685 C0ZK4Q 155535450 EC50 = 284 nM T76685 CGK6Y7 155535538 EC50 = 80 nM T76685 CA6K5I 155535568 Ki = 2 nM T76685 C4TYS3 155535616 EC50 = 21 nM T76685 CF31LR 155535617 EC50 = 120.23 nM T76685 CXTG71 155536120 EC50 = 1113 nM T76685 CMD20W 155536271 Ki = 2600 nM T76685 C3H1VC 155536420 IC50 > 10000 nM T76685 CDQJ85 155536760 EC50 = 1.698 nM T76685 CBK0S3 155536798 EC50 = 234 nM T76685 C7KD3W 155536933 Ki = 1140 nM T76685 CBN0C9 155537341 Ki = 1086 nM T76685 C3TIP1 155537440 EC50 = 58 nM T76685 CI68ZP 155537523 Ki > 40000 nM T76685 CPT5E6 155538176 IC50 > 10000 nM T76685 CQ1PJ9 155538267 Ki = 5 nM T76685 CKM20U 155538552 Ki = 2120 nM T76685 CA2S9E 155538637 EC50 = 3.981 nM T76685 CCL5E1 155538792 Ki > 40000 nM T76685 CB9MN1 155540020 Ki = 6512 nM T76685 C1PBU9 155540079 IC50 = 8 nM T76685 CLFP79 155540709 Ki > 10000 nM T76685 C1DOP8 155540736 EC50 = 730 nM T76685 CKH5R0 155540808 EC50 = 36 nM T76685 C2CA0R 155540863 EC50 = 1150 nM T76685 CJ3MP5 155540943 Ki = 1810 nM T76685 CY5LK9 155541205 Ki = 627 nM T76685 CVRU84 155541432 Ki > 1000 nM T76685 CK0W4A 155541870 EC50 = 1.7 nM T76685 CYW5Z7 155542096 Ki = 3300 nM T76685 CL7NT6 155542142 Ki = 780 nM T76685 C3H2LT 155542283 Ki = 470 nM T76685 C2A8JP 155542531 Ki = 9 nM T76685 CXD78G 155543140 Ki > 10000 nM T76685 CE97SK 155544312 Ki > 10000 nM T76685 CGP4Z6 155544367 IC50 = 4950 nM T76685 C0ER5T 155544651 EC50 = 1100 nM T76685 C1XNB9 155545036 Ki > 10000 nM T76685 C4GE0W 155545108 EC50 > 10000 nM T76685 C7NA0J 155545226 Ki = 500 nM T76685 C6TDM3 155545733 Ki = 6440 nM T76685 C8LD0Y 155545892 Ki = 20 nM T76685 C9QJF1 155546417 Ki = 13 nM T76685 C4E5AY 155546820 Ki = 2.4 nM T76685 C4OFS6 155546920 EC50 = 462 nM T76685 CB1RE9 155547138 Ki = 1.4 nM T76685 CI51BW 155547150 Ki = 3 nM T76685 C9GLF4 155547193 IC50 > 10000 nM T76685 CD7T4W 155547302 Ki > 1000 nM T76685 CM0HZ1 155547797 IC50 = 85 nM T76685 C25LKO 155548028 Ki = 4 nM T76685 CR4WF3 155548082 Ki > 40000 nM T76685 C61JDG 155548443 EC50 = 3100 nM T76685 C9D7IV 155548445 Ki = 518.57 nM T76685 CLT98Z 155548700 IC50 > 10000 nM T76685 C6TPM9 155549206 IC50 > 10000 nM T76685 C83SPR 155549297 EC50 = 35 nM T76685 CFH6B8 155549475 Ki > 1000 nM T76685 CURJ67 155549486 EC50 = 79800 nM T76685 CA8FQ3 155549571 Ki = 1760 nM T76685 C4C0YU 155549576 EC50 = 466 nM T76685 CD31UY 155549880 Ki > 1000 nM T76685 CM9UO8 155549886 IC50 > 10000 nM T76685 CTYX39 155549979 EC50 = 510 nM T76685 C18IUD 155550289 Ki = 903 nM T76685 CPKV56 155550530 Ki > 10000 nM T76685 C73WDS 155551438 EC50 = 1600 nM T76685 CUZ2N8 155551511 IC50 > 10000 nM T76685 CF57LT 155551713 EC50 > 10000 nM T76685 C1S7EG 155551990 IC50 = 5 nM T76685 CR17WN 155552557 Ki = 4 nM T76685 CI57BL 155553206 Ki = 1339.29 nM T76685 C1V2LX 155553407 EC50 = 110 nM T76685 CL9CK6 155553416 EC50 = 191 nM T76685 CV39BX 155553848 EC50 = 17 nM T76685 CAO59L 155553908 Ki = 25 nM T76685 CAG84D 155554628 Ki > 10000 nM T76685 C5YMJ1 155554674 Ki = 64.8 nM T76685 CC9W2O 155555175 IC50 = 4 nM T76685 C5D7BL 155555447 Ki = 1331 nM T76685 CE7N2K 155556020 EC50 = 177 nM T76685 CV59KM 155556037 Ki = 613.7 nM T76685 CHC64Z 155556086 Ki = 860 nM T76685 CRG9D5 155556444 Ki = 380 nM T76685 C8A2ZH 155556549 Ki = 11 nM T76685 CS2G4Q 155556587 Ki > 40000 nM T76685 C06AVX 155557213 EC50 = 992 nM T76685 CD08FU 155557245 Ki = 4 nM T76685 C91JPV 155557850 Ki = 0.11 nM T76685 C5UCL8 155558472 Ki > 10000 nM T76685 C0IOD2 155558946 Ki > 10000 nM T76685 CQ5NT9 155558975 EC50 = 1600 nM T76685 C9J4CP 155559266 Ki = 702.4 nM T76685 C21FEC 155559490 Ki = 4159 nM T76685 C1X2NK 155559788 Ki = 97 nM T76685 CRS6P3 155559856 Ki > 10000 nM T76685 C0S4HQ 155560063 Ki > 40000 nM T76685 C3XL0H 155560208 IC50 > 10000 nM T76685 CKJ7L8 155560630 Ki = 0.9 nM T76685 C4Z7YE 155560703 Ki = 8.2 nM T76685 C72BJQ 155560783 Ki = 0.98 nM T76685 CY52RZ 155560863 IC50 > 10000 nM T76685 C9OJ6V 155561026 IC50 > 10000 nM T76685 CI6QS0 155561427 EC50 = 1100 nM T76685 C27XCM 155561507 Ki = 54.4 nM T76685 C9VWA7 155561675 Ki > 1000 nM T76685 CS8G1A 155561709 Ki > 10000 nM T76685 CSZ64Y 155562059 EC50 = 40 nM T76685 CX4H8P 155562737 Ki > 1000 nM T76685 CU56LB 155562889 EC50 = 489.78 nM T76685 C84VUF 155563880 Ki = 593 nM T76685 C5C6ZE 155564195 Ki = 17 nM T76685 CH7KX9 155564385 Ki = 1482 nM T76685 CNS30G 155564805 Ki = 272 nM T76685 C3B9RS 155564863 IC50 > 10000 nM T76685 C2EQD9 155565124 EC50 > 10000 nM T76685 CHC63R 155565172 Ki = 395 nM T76685 C18MHX 155565431 Ki = 1.1 nM T76685 CG26YT 155565779 Ki = 0.6 nM T76685 CSC45B 155566194 Ki > 10000 nM T76685 C2NB9W 155566555 Ki = 430 nM T76685 CXKJ16 155566978 IC50 > 10000 nM T76685 C3AWZ5 155567068 Ki = 15.4 nM T76685 C2FOQ9 155567428 IC50 > 10000 nM T76685 C1SYW9 155567786 Ki = 6.3 nM T76685 CRV96F 155567845 EC50 = 22 nM T76685 CF7L0T 155568163 Ki = 332.6 nM T76685 CGQT89 155568550 Ki = 218.1 nM T76685 C9R2HS 155568851 Ki > 10000 nM T76685 CH89DI 155569209 Ki = 1 nM T76685 CA5V2O 155569605 EC50 > 10000 nM T76685 CP9TR0 10324985 Ki > 10000 nM T76685 C13REG 44471685 Ki = 3.4 nM T76685 C6MWP8 46880677 Ki > 1000 nM T76685 C70OFQ 46880728 Ki > 1000 nM T76685 C8NPM1 46905057 Ki = 1470 nM T76685 C8AJN0 46916610 Ki = 10000 nM T76685 D00UZO 5712057 Ki = 912 nM T76685 D00VCW 5311006 Ki = 5.3 nM T76685 D01DIT 5283446 Ki > 41400 nM T76685 D01JHA 44431964 Ki = 5.2 nM T76685 D01MCD 25059294 IC50 = 3 nM T76685 D01PEC 24995603 IC50 = 0.2 nM T76685 D01PZU 44440707 Ki = 2381 nM T76685 D01RWS 16066912 Ki > 10000 nM T76685 D01VIA 994313 Ki = 164 nM T76685 D01ZHW 5283389 Ki > 10000 nM T76685 D02GOH 6604822 Ki = 1500 nM T76685 D02INF 5311216 Ki = 4888 nM T76685 D02NAW 24995605 IC50 = 0.7 nM T76685 D02POA 11551123 Ki = 23 nM T76685 D02SMK 1172084 EC50 > 30000 nM T76685 D02VSL 6918505 Ki = 0.797 nM T76685 D03HFM 42617984 Ki = 11 nM T76685 D03RFS 1293167 Ki = 560 nM T76685 D03SCD 44448616 Ki > 10000 nM T76685 D03TPB 11498260 Ki = 750 nM T76685 D04AMC 11559610 Ki = 3900 nM T76685 D04DQJ 72303 Ki = 6.46 nM T76685 D04ECZ 42617986 Ki = 570 nM T76685 D04GDY 638026 Ki = 28.5 nM T76685 D04ICJ 1358608 Ki = 52 nM T76685 D05DFO 44406102 Ki = 1500 nM T76685 D05QPE 5282272 Ki = 53.4 nM T76685 D05QTX 44828492 EC50 = 9.05 nM T76685 D05RGU 44406075 Ki = 300 nM T76685 D05TQX 11702887 Ki > 10000 nM T76685 D05ZUX 44207909 Ki >= 1000 nM T76685 D06DTC 24995604 IC50 = 0.4 nM T76685 D06EHU 11406508 Ki = 1379 nM T76685 D06GAF 2836828 Ki > 50 nM T76685 D06JBN 5282280 EC50 = 23 nM T76685 D06JFN 1076739 Ki > 1000 nM T76685 D06NXC 24996886 IC50 = 0.7 nM T76685 D06RIK 44406076 Ki = 1000 nM T76685 D06SRX 135743701 EC50 = 867 nM T76685 D06YQD 44440709 Ki = 178 nM T76685 D07MBC 5283454 Ki = 1100 nM T76685 D08BNY 44406107 Ki = 4900 nM T76685 D08DOG 25130235 Ki > 10000 nM T76685 D08DZK 44406080 Ki = 600 nM T76685 D08GLU 44431968 Ki = 320 nM T76685 D08JYT 6483057 Ki = 20 nM T76685 D08MON 16067266 Ki >= 10000 nM T76685 D08OAQ 44431961 Ki = 91 nM T76685 D08TXL 11584525 IC50 = 330 nM T76685 D08UKF 44406087 Ki = 5400 nM T76685 D08VLG 11290338 Ki = 1.7 nM T76685 D08YQT 2125 IC50 = 0.32 nM T76685 D09BYO 24996885 IC50 = 1.7 nM T76685 D09CKZ 9799945 Ki = 6.8 nM T76685 D09DSK 9799540 Ki = 1.2 nM T76685 D09FMK 4302963 Ki = 840 nM T76685 D09KFJ 44581105 Ki = 3134 nM T76685 D09RIC 46203026 IC50 = 6000 nM T76685 D0A2KW 44421550 Ki = 2900 nM T76685 D0A9PS 5281969 Ki = 11 nM T76685 D0B8EP 11524275 EC50 = 1050 nM T76685 D0B8GY 44440706 Ki = 3848 nM T76685 D0BS7G 5311215 Ki = 1043 nM T76685 D0CO6T 11386747 IC50 = 7.5 nM T76685 D0D6OH 104895 IC50 = 0.13 nM T76685 D0D7OR 44593431 Ki = 5.26 nM T76685 D0D8PZ 93147 Ki = 75.4 nM T76685 D0E0AA 24996566 IC50 = 46 nM T76685 D0E3ET 9950486 Ki = 400 nM T76685 D0E9HC 44421549 Ki = 7050 nM T76685 D0EC6B 6443006 Ki = 1940 nM T76685 D0F3CH 11233636 Ki > 10000 nM T76685 D0F4BE 11508826 Ki = 3500 nM T76685 D0F4BX 9821569 Ki = 0.06 nM T76685 D0FF6S 16038374 IC50 = 10000 nM T76685 D0FJ1I 46891225 IC50 = 1.7 nM T76685 D0G2EQ 42617990 Ki = 28 nM T76685 D0G3TV 2440433 EC50 > 30000 nM T76685 D0G4VV 9893254 Ki = 1.3 nM T76685 D0G7GF 44431966 Ki = 15 nM T76685 D0H1DV 10215860 IC50 = 326 nM T76685 D0H6DL 11609579 Ki = 6296 nM T76685 D0I1OJ 44406101 Ki = 6400 nM T76685 D0I4AF 24992105 IC50 = 2.1 nM T76685 D0J3XJ 44578696 Ki = 1900 nM T76685 D0J5KA 44406095 Ki = 3700 nM T76685 D0J7CR 42617983 Ki = 14 nM T76685 D0J8KW 3081355 Ki = 2 nM T76685 D0K4PV 46891372 IC50 = 1.8 nM T76685 D0K5DA 11502240 Ki = 500 nM T76685 D0K7QP 44591633 Ki = 1400 nM T76685 D0K8MN 44448617 Ki = 1600 nM T76685 D0L1UA 10811495 Ki = 200 nM T76685 D0L6RT 56463 IC50 = 453 nM T76685 D0LX4U 11576518 Ki = 1800 nM T76685 D0N0ME 2809754 Ki = 239 nM T76685 D0O3NY 10141893 Ki = 280 nM T76685 D0O4LO 23654364 Ki = 12.9 nM T76685 D0O7ZJ 11461586 Ki = 1054 nM T76685 D0OQ5H 46891330 IC50 = 3.7 nM T76685 D0P5VJ 10248110 Ki = 12.3 nM T76685 D0PC5A 44243144 Ki = 560 nM T76685 D0PE8U 25178128 Ki = 300 nM T76685 D0Q0XV 44591632 Ki = 820 nM T76685 D0Q4DB 5282273 Ki = 34.4 nM T76685 D0Q8QH 11638703 Ki > 10000 nM T76685 D0Q9GU 1792197 EC50 > 30000 nM T76685 D0R1UA 3137700 Ki > 50 nM T76685 D0R6MB 46891274 IC50 = 97 nM T76685 D0R7QF 42617989 Ki = 20 nM T76685 D0R9VY 24992763 IC50 = 14 nM T76685 D0T2RY 9948320 Ki >= 1000 nM T76685 D0T3CP 11645841 Ki > 10000 nM T76685 D0T4SE 44406097 Ki = 2400 nM T76685 D0U3ME 44300692 Ki > 30000 nM T76685 D0U5LL 2543 Ki = 13 nM T76685 D0UD9H 4302962 Ki = 13.2 nM T76685 D0V0YM 24871527 EC50 = 5.8 nM T76685 D0V2NQ 2385541 Ki = 3400 nM T76685 D0X8FV 44440708 Ki = 656 nM T76685 D0Y1MM 11710300 Ki = 470 nM T76685 D0Z1NH 42617985 Ki = 600 nM T76685 D0Z5CX 4225440 Ki = 58 nM T76685 D0Z7OB 44406064 Ki = 2800 nM T76685 D0Z9GI 11552795 Ki = 2900 nM T76685 D0ZM1T 44250208 Ki = 7 nM T76685 D0ZU9Z 5311257 Ki = 141 nM T17552 D0E3TC 44259 IC50 = 36.3 nM T17552 D03BNU 59604787 IC50 > 10000 nM T17552 D0T3ME 156422 IC50 > 30000 nM T17552 CI51GR 370373 IC50 = 170 nM T17552 CP3J8Y 867021 IC50 > 10000 nM T17552 CXZK10 3162043 IC50 = 280 nM T17552 CU5HA2 3163413 IC50 = 160 nM T17552 C58OZW 3578433 IC50 > 10000 nM T17552 CN4B7P 5019834 IC50 = 980 nM T17552 C5O2NF 7161416 IC50 = 7300 nM T17552 CIG04V 7186151 IC50 = 300 nM T17552 CR1H5X 7186158 IC50 = 150 nM T17552 CSZO42 53245473 IC50 = 11 nM T17552 CF1B2M 53347948 IC50 > 10000 nM T17552 C9WUH8 53347978 IC50 > 10000 nM T17552 CFB93A 53347979 IC50 = 76 nM T17552 C4XV3U 53347999 IC50 = 580 nM T17552 CR47DL 53377411 IC50 = 270 nM T17552 CD51HW 53377418 IC50 = 380 nM T17552 C31LNY 53377419 IC50 = 78 nM T17552 CR68JP 53377420 IC50 = 530 nM T17552 CV32AS 53377429 IC50 = 110 nM T17552 CG8PU3 53377430 IC50 = 1600 nM T17552 CH5E9N 53377431 IC50 = 1600 nM T17552 C6Y5DA 53377438 IC50 = 250 nM T17552 CA1F2V 53377442 IC50 = 410 nM T17552 CPNS41 53377443 IC50 > 10000 nM T17552 CZHE94 53377446 IC50 = 1600 nM T17552 CHFE05 53377447 IC50 > 10000 nM T17552 CA58WB 53377448 IC50 = 14 nM T17552 C25YJF 53377455 IC50 = 4000 nM T17552 C8NA4L 53384644 IC50 > 30000 nM T17552 CV63UL 67240318 IC50 > 10000 nM T17552 C2MD1Q 155513187 IC50 > 10000 nM T17552 D00ERW 44444843 Ki > 1638 nM T17552 D01TDV 71452170 IC50 = 7 nM T01007 D0I6LH 107985 IC50 = 14 nM T01007 D05VXK 56848369 IC50 = 77000 nM T01007 D0CM5P 6737869 IC50 = 34000 nM T01007 D0Z4SW 56848967 IC50 = 243000 nM T01007 CZQF03 9589606 EC50 = 199.53 nM T01007 CH0JQ4 9696680 EC50 = 6309.57 nM T01007 CJ79ZS 9831050 EC50 = 4200 nM T01007 C8TRG1 9950925 IC50 = 5000000 nM T01007 CNY07E 10149969 IC50 = 67800 nM T01007 CI16WO 10232703 EC50 = 28183.83 nM T01007 C2BTQ1 10395438 EC50 = 25.12 nM T01007 CC41EQ 10483914 EC50 = 3000 nM T01007 CP1N9D 11557006 Ki = 600 nM T01007 CTO42L 25108278 EC50 = 30 nM T01007 CZO38G 25108279 EC50 = 7943.28 nM T01007 CJY10U 25108280 EC50 = 10000 nM T01007 CYN0U4 25108338 EC50 = 2511.89 nM T01007 CH27QL 25108339 EC50 = 125.89 nM T01007 CMWE08 25108340 EC50 = 25.12 nM T01007 C83RMZ 25108341 EC50 = 6309.57 nM T01007 CL6K2Z 25108342 EC50 = 50.12 nM T01007 C29JGO 44433860 EC50 = 700 nM T01007 CX1VT3 44433864 EC50 = 1000 nM T01007 CC19MI 44433865 EC50 = 1800 nM T01007 CK4U1Y 44433867 EC50 = 1900 nM T01007 C7O2NA 44433868 EC50 = 1100 nM T01007 CNI8S7 44433869 EC50 = 400 nM T01007 CC2X4D 44433871 EC50 = 900 nM T01007 CS6J3Z 44433872 EC50 = 500 nM T01007 CYTF75 44433873 EC50 = 600 nM T01007 CUB3R9 44433874 EC50 = 600 nM T01007 CASU09 44433875 EC50 = 2500 nM T01007 C2F4XC 44433877 EC50 = 1300 nM T01007 CPR27Y 44433878 EC50 = 5000 nM T01007 CI5CM4 44433880 EC50 = 3000 nM T01007 CZYW46 44433883 EC50 = 2800 nM T01007 CF90JN 44433885 EC50 = 1400 nM T01007 C9YA2Q 44433886 EC50 = 300 nM T01007 CKH5P3 44433887 EC50 = 1300 nM T01007 CQTL72 44433892 EC50 = 3300 nM T01007 C39BRL 44433894 EC50 = 1700 nM T01007 C7DCM0 44433900 EC50 = 300 nM T01007 C6T2VJ 44433902 EC50 = 160 nM T01007 CWX82D 44433903 EC50 = 100 nM T01007 C8W3KA 44433904 EC50 = 100 nM T01007 C67QDB 44433905 EC50 = 100 nM T01007 C0AW2I 44433906 EC50 = 590 nM T01007 C2Z5HR 44433907 EC50 = 14900 nM T01007 C78DSJ 44433908 EC50 = 15800 nM T01007 CNIS69 44433909 EC50 = 4800 nM T01007 C4FJ3Y 44433910 EC50 = 10300 nM T01007 CJA36H 44433911 EC50 = 800 nM T01007 COT1X0 44433912 EC50 = 100 nM T01007 CW3N9A 44433913 EC50 = 100 nM T01007 CVTD69 44433914 EC50 = 100 nM T01007 CNP5D4 44433915 EC50 = 1600 nM T01007 C8F2YR 44433916 EC50 = 100 nM T01007 CJ0H1W 44433917 EC50 = 100 nM T01007 CF6NY1 44433918 EC50 = 4300 nM T01007 CT9RV0 44433940 EC50 = 200 nM T01007 C98REM 44433947 EC50 = 170 nM T01007 CC25TI 44433948 EC50 = 600 nM T01007 C3FK7I 44433949 EC50 = 320 nM T01007 CKXO16 44433963 EC50 = 1200 nM T01007 CFK1A0 44433964 EC50 = 1000 nM T01007 CCNA17 44433965 EC50 = 1100 nM T01007 CQ6Z4N 44433966 EC50 = 2000 nM T01007 C5VZ8G 44433967 EC50 = 600 nM T01007 C04RTO 44433968 EC50 = 1200 nM T01007 CCH60Z 44433970 EC50 = 1200 nM T01007 CGP93I 44433971 EC50 = 3600 nM T01007 C78NPU 49788150 EC50 > 50000 nM T01007 CH14XL 49788153 EC50 > 100000 nM T01007 CL5A8W 49788154 EC50 > 4000 nM T01007 CMC39J 49788155 EC50 > 100000 nM T01007 CGV0Q5 49788311 EC50 = 199.53 nM T01007 C3VNW4 49788378 EC50 = 12589.25 nM T01007 CBL79Q 49788379 EC50 > 50000 nM T01007 C9NM2I 49788380 EC50 = 316.23 nM T01007 CWXQ13 49788381 EC50 = 1000 nM T01007 CU5K0J 49788439 EC50 = 408 nM T01007 CA14BD 49788440 EC50 = 1995.26 nM T01007 C4Q3EK 49788441 EC50 = 7100 nM T01007 CY9X3A 49788504 EC50 = 12589.25 nM T01007 C02BPK 49788505 IC50 = 57000 nM T01007 CP4W7E 49788574 IC50 = 2000 nM T01007 C45UPM 51351273 EC50 = 142 nM T01007 CC5ES7 51351274 EC50 = 311 nM T01007 C4KPY5 51351408 EC50 = 3500 nM T01007 C8FCZ1 51351409 EC50 = 6590 nM T01007 C0P5FT 52948093 EC50 = 6100 nM T01007 C36PSZ 53318281 IC50 = 690 nM T01007 CUN9P6 53326692 EC50 = 138 nM T01007 CH4FR9 54582896 EC50 = 1400 nM T01007 CD86HV 56639666 IC50 = 400 nM T01007 C8UT1Y 56640042 EC50 = 1995.26 nM T01007 CLE0S5 56640398 IC50 = 8600 nM T01007 C2AW5B 56640474 IC50 = 1900 nM T01007 CY63EN 56640547 IC50 = 1200 nM T01007 C1U8GS 56640610 EC50 = 700 nM T01007 CDT76U 56640611 EC50 = 700 nM T01007 CESI03 57330164 IC50 = 1100 nM T01007 CNEO43 71511553 IC50 = 1258.93 nM T01007 CXB78U 73346321 EC50 = 200 nM T01007 CA41PT 73347818 IC50 = 700000 nM T01007 C7NTU0 73355411 EC50 = 4 nM T01007 CZO78P 117977940 IC50 = 4.8 nM T01007 CTH0N8 117978042 IC50 = 2 nM T01007 CSQ7N6 117990832 IC50 = 4400 nM T01007 CD21PQ 117991137 IC50 = 2 nM T01007 C0UDR9 126961334 IC50 = 4200 nM T01007 CW03MF 126961335 IC50 < 2.5 nM T01007 CO6M2S 127035718 Ki = 1940 nM T01007 C14WCD 127035910 Ki = 627 nM T01007 C8MOC4 127036298 IC50 = 2800 nM T01007 C3MTV5 127036301 IC50 > 10000 nM T01007 C8MC6H 134137699 IC50 = 8900 nM T01007 CY8N3X 134143255 IC50 = 3100 nM T01007 C9CS4G 134147747 EC50 = 700 nM T01007 C6BSE1 137633152 EC50 = 398.11 nM T01007 CS9UM8 137637330 EC50 = 199.53 nM T01007 CPXI31 137638214 EC50 = 95 nM T01007 C6W5BL 137641156 EC50 = 62 nM T01007 CJ8EN5 137643158 EC50 > 100000 nM T01007 CZ2W3S 137650859 EC50 > 100000 nM T01007 CD25WP 137653967 EC50 = 79.43 nM T01007 CW4D2N 137654325 EC50 = 31.62 nM T01007 C3V9ZC 137654661 EC50 = 79.43 nM T01007 C9F1TA 137661916 EC50 = 18 nM T01007 CA8EX2 145962815 IC50 = 6000 nM T01007 CPX6Q0 155512671 IC50 > 50000 nM T01007 C2ORE8 155534488 IC50 = 2 nM T01007 CQN9L7 155536026 IC50 > 50000 nM T01007 CFDM94 155549751 IC50 = 3300 nM T01007 CN4WT6 155564785 IC50 > 50000 nM T01007 CENS94 155567301 IC50 = 860 nM T01007 CYSM34 44433870 EC50 = 400 nM T57291 D01SLG 446512 IC50 = 0.07 nM T57291 D0O1BJ 445434 IC50 = 0.1 nM T57291 D0O7ZE 5311365 IC50 = 0.13 nM T52189 CIU6R4 442729 IC50 = 12600 nM T52189 C1U2AF 1187307 IC50 = 11900 nM T52189 C5UJF1 1637033 IC50 = 4100 nM T52189 CJR68K 2355050 IC50 = 13800 nM T52189 C48NWG 10251951 IC50 = 2900 nM T52189 CD25XZ 10267060 IC50 = 9600 nM T52189 CWR52Q 10497365 Ki = 320000 nM T52189 C9E6IL 10501796 Ki = 13000 nM T52189 CI37QA 10502374 Ki = 550 nM T52189 CP2BT9 10526128 Ki = 26000 nM T52189 C2N0VW 10527433 Ki = 710 nM T52189 CTS70W 10527606 Ki = 2900 nM T52189 C5P1LF 10573701 Ki = 9500 nM T52189 CTBM54 10620844 Ki = 41000 nM T52189 C3F5IA 10622175 Ki = 620 nM T52189 CH2J1D 10624056 Ki = 300 nM T52189 CV6Y4S 10645065 Ki = 5700 nM T52189 C7V3DY 10647160 Ki = 750 nM T52189 C9L4EW 10669261 Ki = 121000 nM T52189 C6QGW3 10669850 Ki = 18000 nM T52189 CI6LO0 10671758 Ki = 2700 nM T52189 C72BSJ 10673460 Ki = 21000 nM T52189 CY59WJ 10692511 Ki = 19000 nM T52189 COAF46 10712724 Ki = 300000 nM T52189 C0LDZ7 10741647 Ki = 3900 nM T52189 CM2F9L 10743119 Ki = 11000 nM T52189 CIS6T4 10743296 Ki = 5100 nM T52189 CVI34J 10765158 Ki = 1800 nM T52189 COQ0T9 10766613 Ki = 300 nM T52189 CM3J8C 10767318 Ki = 2900 nM T52189 C9RH2Z 10787020 Ki = 3500 nM T52189 C3F8LP 10790840 Ki = 1100 nM T52189 C8MVO9 10811352 Ki = 2000 nM T52189 CNOF13 10811591 Ki = 3200 nM T52189 CLKO57 10814072 Ki = 2700 nM T52189 C9KL8D 10814362 Ki = 370 nM T52189 C6FTS8 10814676 Ki = 5000 nM T52189 CIFC12 11794391 Ki = 160000 nM T52189 CZ38RO 11797483 Ki = 64000 nM T52189 C14KRF 16747776 IC50 = 442 nM T52189 CM23OT 44346088 Ki = 220 nM T52189 CGM2L7 44442231 IC50 = 1100 nM T52189 CWZ7X3 44442234 IC50 = 2300 nM T52189 C2QT3O 44442236 IC50 = 7600 nM T52189 CW3VQ6 44442239 IC50 = 5600 nM T52189 C7K3DH 44442242 IC50 = 190 nM T52189 CO1AK5 44442284 IC50 = 6900 nM T52189 C7F4JQ 44442285 IC50 = 10900 nM T52189 CRK5B3 44442286 IC50 = 8100 nM T52189 CWT93Q 44442287 IC50 = 370 nM T52189 CKY4H6 44442288 IC50 = 340 nM T52189 CQ2WM1 57316190 Ki = 620 nM T52189 CLVK63 60152136 IC50 = 7500 nM T52189 C63VKQ 71449783 Ki = 710 nM T52189 CK2US5 71449784 Ki = 220 nM T52189 C0JQ7M 71458796 Ki = 700 nM T52189 CAXW52 71460614 Ki = 3200 nM T52189 CWCF61 71462317 Ki = 370 nM T52189 C3RTZ1 102204395 IC50 = 25800 nM T52189 CN90WH 135466913 IC50 = 7000 nM T52189 CW8I7A 137638038 IC50 = 13300 nM T52189 C3GH6K 137638701 IC50 = 29700 nM T52189 CB9MN0 137647084 IC50 = 3800 nM T52189 CG7AC0 137647506 IC50 = 23500 nM T52189 C6ARJ3 137653432 IC50 = 21100 nM T52189 C1T5GC 137654084 IC50 = 30000 nM T52189 C1KN8F 137657464 IC50 = 21200 nM T52189 CH2SF9 137657898 IC50 = 18800 nM T52189 CB2I5V 155517051 IC50 = 2800 nM T52189 C1HL4K 155519234 IC50 = 2800 nM T52189 C2WP6O 155522824 IC50 = 2800 nM T52189 CW1V5X 155522892 IC50 = 2800 nM T52189 D09AXB 10835222 Ki = 770 nM T52189 D0IC1N 185620 IC50 = 150 nM T64682 D0EG1I 9926791 IC50 > 10000 nM T64682 D01NEC 51042438 IC50 = 211 nM T64682 D0E3TC 44259 IC50 = 6.75 nM T64682 D03BNU 59604787 IC50 > 10000 nM T64682 D02GEJ 5326976 IC50 = 3570 nM T64682 D04FHB 6918852 Ki > 5000 nM T64682 D0T3ME 156422 IC50 > 30000 nM T64682 CAV19R 2360773 IC50 > 10000 nM T64682 C04IXB 2958682 IC50 = 60000 nM T64682 CIAL53 9819282 IC50 > 250000 nM T64682 CW8V0K 9864418 IC50 > 33000 nM T64682 CM5Z8X 9869943 IC50 > 1000 nM T64682 C2TC1L 9910609 IC50 > 125000 nM T64682 CJO47T 9948405 IC50 > 10000 nM T64682 C37GXK 9983303 IC50 > 33000 nM T64682 CV8I5X 9999342 IC50 > 10000 nM T64682 CJX43Z 10055074 IC50 > 50000 nM T64682 C2C1BP 10089048 IC50 > 33000 nM T64682 CLP79V 10196532 IC50 > 50000 nM T64682 C0R5AX 10215912 IC50 > 50000 nM T64682 C8V6RI 10240275 IC50 > 50000 nM T64682 C5TQ7X 10247543 IC50 > 10000 nM T64682 C4MOF8 10312133 IC50 > 50000 nM T64682 CAK9U4 10415819 IC50 > 50000 nM T64682 C2WQ8M 10473563 IC50 > 10000 nM T64682 CRX6F0 10479082 IC50 > 33000 nM T64682 CBOP58 11293798 Ki > 10000 nM T64682 C26BZX 11362471 Ki > 10000 nM T64682 C43NPS 11373886 IC50 > 10000 nM T64682 CWXB93 11397177 Ki > 10000 nM T64682 CWM18I 11406175 IC50 > 50000 nM T64682 C1WXC5 11417488 IC50 > 50000 nM T64682 C0APW4 11422034 IC50 = 10000 nM T64682 C64IGY 11448608 Ki > 5000 nM T64682 C0H6QS 11495680 IC50 > 10000 nM T64682 CIW9L5 11502867 IC50 > 10000 nM T64682 CK2Q0X 11516978 IC50 > 10000 nM T64682 C2BH1E 11524857 IC50 = 261 nM T64682 CPE53F 11526238 IC50 > 10000 nM T64682 C5BM4T 11531799 IC50 > 10000 nM T64682 C53OSD 11532048 IC50 > 10000 nM T64682 CC4QM5 11532676 IC50 > 10000 nM T64682 CTG83F 11539329 Ki > 9400 nM T64682 CE5H7D 11544170 IC50 = 1300 nM T64682 C01FVM 11546457 IC50 > 10000 nM T64682 CACS26 11561968 Ki > 2000 nM T64682 CNBM81 11562171 IC50 > 10000 nM T64682 C45QDX 11568147 IC50 = 2200 nM T64682 CMIL86 11590363 Ki > 9400 nM T64682 C0NV9Y 11596881 IC50 > 10000 nM T64682 C1BLZ5 11620055 IC50 > 10000 nM T64682 C9T6SC 11640926 Ki > 9400 nM T64682 C24GRQ 11661959 IC50 > 10000 nM T64682 C7XEV0 11664023 IC50 > 50000 nM T64682 CS72ED 11682843 IC50 > 10000 nM T64682 CU0E8O 11690457 Ki > 2000 nM T64682 CLC53E 11691173 IC50 > 10000 nM T64682 CB0AP2 11705863 Ki > 2000 nM T64682 C1FTX3 11719305 IC50 > 10000 nM T64682 CB2Q7D 11952989 IC50 = 880 nM T64682 C9LOP1 11953177 IC50 = 400 nM T64682 CSA02I 15979148 IC50 > 50000 nM T64682 CBE54Y 15979149 IC50 > 50000 nM T64682 C92FEN 15979151 IC50 > 50000 nM T64682 C9QO8U 15979276 IC50 > 50000 nM T64682 CFPW41 16007116 Ki > 9400 nM T64682 C9TU1O 16046126 IC50 > 1000 nM T64682 CBM80K 16091080 IC50 > 50000 nM T64682 C5VPH9 16129448 IC50 = 606 nM T64682 CVS0T5 17754396 IC50 > 10000 nM T64682 C5AR9M 21103197 IC50 > 50000 nM T64682 CG6D4M 23647319 IC50 > 10000 nM T64682 CY8Z7X 23647330 IC50 > 10000 nM T64682 C4XD8H 23647348 IC50 > 10000 nM T64682 C7YG1N 24759534 IC50 = 27 nM T64682 C61KPI 24856363 IC50 > 33000 nM T64682 CO42DC 44138048 IC50 > 10000 nM T64682 CL65QV 44138049 IC50 > 10000 nM T64682 CV09DY 44410717 IC50 > 10000 nM T64682 CP3CI1 44410720 IC50 > 10000 nM T64682 C8W7AD 44410723 IC50 > 10000 nM T64682 CAT5X4 44410829 IC50 > 10000 nM T64682 CC6Y5P 44410844 IC50 > 10000 nM T64682 CG34TY 44410851 IC50 > 10000 nM T64682 C41EIA 44410869 IC50 > 10000 nM T64682 CB6AE8 44410948 IC50 > 10000 nM T64682 CXZG12 44410949 IC50 > 10000 nM T64682 CS7IE9 44410953 IC50 > 10000 nM T64682 CA9M4X 44410954 IC50 > 10000 nM T64682 C3SP5H 44410955 IC50 > 10000 nM T64682 C5D6YP 44410956 IC50 > 10000 nM T64682 C5W1VC 44410959 IC50 > 10000 nM T64682 CM1C2G 44410960 IC50 > 10000 nM T64682 CVSI80 44411048 IC50 > 10000 nM T64682 CN72BR 44411161 IC50 > 10000 nM T64682 C4AW0O 44411183 IC50 > 10000 nM T64682 CETQ79 44427518 IC50 > 50000 nM T64682 COPG94 44427519 IC50 > 10000 nM T64682 CZ9L8F 44572052 IC50 > 50000 nM T64682 CIV48S 44572053 IC50 > 50000 nM T64682 CFVA91 44572054 IC50 > 50000 nM T64682 CZE8M9 44572055 IC50 > 50000 nM T64682 C7Q1VU 44580077 IC50 > 33000 nM T64682 CL90SE 44580358 IC50 > 33000 nM T64682 CK1VE7 44580420 IC50 > 33000 nM T64682 CH2R7X 44580449 IC50 > 33000 nM T64682 C1VH0C 44580532 IC50 = 32000 nM T64682 CXC52J 44580649 IC50 > 33000 nM T64682 CE32BQ 44580689 IC50 > 33000 nM T64682 C8Z5AX 44580778 IC50 > 33000 nM T64682 C3WA1X 45267446 IC50 = 5000 nM T64682 COFN91 45268287 IC50 = 3160 nM T64682 CBW2Y1 45268295 IC50 = 160 nM T64682 C04CMT 45268304 IC50 = 63 nM T64682 CH4B1K 45270042 IC50 = 5 nM T64682 CSEA01 45271705 IC50 = 20 nM T64682 C3A5NY 45272590 IC50 = 50 nM T64682 C7JB0X 45273462 IC50 = 125 nM T64682 C1IR7Y 45273473 IC50 = 40 nM T64682 CZ58FY 46215814 IC50 > 10000 nM T64682 CY3HW5 46224684 IC50 = 690 nM T64682 CLS29B 46872626 IC50 > 10000 nM T64682 C2O8RZ 46886323 IC50 > 1000 nM T64682 CHSF07 49806372 IC50 > 1000 nM T64682 CEQN27 52936621 Ki > 1000 nM T64682 C8NA4L 53384644 IC50 = 19000 nM T64682 C8W6IG 57395117 IC50 > 30000 nM T64682 CXJ63M 59603829 IC50 = 63 nM T64682 CQEU96 59603842 IC50 = 200 nM T64682 COH62U 60097413 IC50 > 10000 nM T64682 C1MR8Q 60097495 IC50 > 10000 nM T64682 CV63UL 67240318 IC50 > 10000 nM T64682 C5DGR9 69036886 IC50 = 10000 nM T64682 CH0B8N 70789756 IC50 > 30000 nM T64682 CKT60L 71455860 Ki = 260 nM T64682 CCV93P 71506845 IC50 = 1 nM T64682 CNRQ28 71534719 IC50 = 2 nM T64682 C4FN3C 71534721 IC50 = 2 nM T64682 CRU94Y 71536970 IC50 = 3 nM T64682 C4JAS9 71537258 IC50 = 439 nM T64682 CQ0P6A 71537259 IC50 = 496 nM T64682 CS4P8Z 71537260 IC50 = 419 nM T64682 C6G2WE 71537261 IC50 = 5 nM T64682 CN23CP 71537262 IC50 = 639 nM T64682 C43CDG 71537263 IC50 = 2 nM T64682 C1QVR4 71537540 IC50 = 2 nM T64682 CG95ZA 71537541 IC50 = 3 nM T64682 C8RMV5 71537542 IC50 = 2 nM T64682 CT24GH 71537543 IC50 = 605 nM T64682 CQ92BN 71537544 IC50 = 4 nM T64682 CU5PQ7 71537545 IC50 = 3 nM T64682 CT8A0P 71537834 IC50 = 580 nM T64682 CBG1I5 71537835 IC50 = 2 nM T64682 CW8U2R 71537836 IC50 = 2 nM T64682 CTNA59 71537837 IC50 = 3 nM T64682 C7N2QU 71537838 IC50 = 2 nM T64682 CPI7Y1 71537839 IC50 = 2 nM T64682 CL0C9R 71538111 IC50 = 10 nM T64682 CKL9R3 71538112 IC50 = 183 nM T64682 C4O9XW 71538663 IC50 = 16 nM T64682 CP6J8H 71538952 IC50 = 2 nM T64682 CZA91T 71538955 IC50 = 407 nM T64682 CA3O6K 71552696 IC50 > 30000 nM T64682 C1NPL0 71552941 IC50 > 30000 nM T64682 CA4PS8 71552942 IC50 > 30000 nM T64682 C0DL3F 72698602 IC50 = 5 nM T64682 CG3KC8 86268372 IC50 < 1.5 nM T64682 C3SK2U 89463862 IC50 = 910 nM T64682 CX56FT 89464020 IC50 = 21 nM T64682 C16MEP 89464440 IC50 = 1490 nM T64682 C8YQE2 89464503 IC50 = 15 nM T64682 C1HW4B 89735655 IC50 = 810 nM T64682 C0VGI3 90421307 IC50 < 1.2 nM T64682 CW6FD3 90421822 IC50 < 1.2 nM T64682 C8ZMX4 118720597 IC50 < 1.5 nM T64682 C7LSK8 118720598 IC50 < 1.2 nM T64682 C0K9GY 118720599 IC50 < 1.5 nM T64682 C6SBU0 118720600 IC50 = 1.5 nM T64682 C6I3NB 118720601 IC50 = 150 nM T64682 CV1QZ2 118720602 IC50 = 6.2 nM T64682 CVH78B 118720603 IC50 = 130 nM T64682 C0UKZ7 118720604 IC50 = 390 nM T64682 CR58YZ 118721247 IC50 = 7140 nM T64682 C94SUJ 118721248 IC50 = 2260 nM T64682 C7AFT2 118721249 IC50 = 1800 nM T64682 C0BCF3 118721250 IC50 = 315 nM T64682 CH7T9W 118721251 IC50 = 28 nM T64682 CV26CL 118721252 IC50 = 13200 nM T64682 CUWC81 118721253 IC50 = 3 nM T64682 CG69KJ 118721254 IC50 = 14 nM T64682 CQ2TS0 118721255 IC50 = 6840 nM T64682 CTCO24 118721256 IC50 < 1 nM T64682 C2C3VM 118721257 IC50 = 9720 nM T64682 CCU57B 118721258 IC50 < 1 nM T64682 CZCK14 118721259 IC50 < 1 nM T64682 CC9E8N 118721260 IC50 = 199 nM T64682 CYS24W 118721261 IC50 = 46 nM T64682 C3IQA4 118721262 IC50 < 2 nM T64682 C0MID8 118721263 IC50 = 1 nM T64682 C2WC8M 118721264 IC50 < 1 nM T64682 CT35IM 118721265 IC50 = 9 nM T64682 C6F0EY 118721266 IC50 < 1 nM T64682 C6U7EN 118721271 IC50 < 1 nM T64682 CSX65L 118721272 IC50 = 4760 nM T64682 CJ9P6X 118721273 IC50 = 29 nM T64682 CU60YC 135431661 IC50 = 290 nM T64682 C62DAQ 135489099 IC50 = 138 nM T64682 CRJ45X 135589980 IC50 = 1320 nM T64682 C0J3BN 135678111 IC50 = 1500 nM T64682 C26ESH 136060555 IC50 = 15000 nM T64682 CI1E8V 137634241 IC50 > 10000 nM T64682 CC73PA 138911338 IC50 = 145 nM T64682 C6VB3O 145925651 IC50 >= 5000 nM T64682 CSU93V 155077019 IC50 = 102 nM T64682 C2MD1Q 155513187 IC50 > 10000 nM T64682 CL5DR0 155525783 IC50 = 59 nM T64682 D00ERW 44444843 Ki = 8176 nM T64682 D00HVA 11624601 Ki > 9400 nM T64682 D07ADX 54764565 IC50 = 201 nM T64682 D09XIL 11396738 IC50 > 125000 nM T64682 D0A7FQ 11644425 IC50 = 2700 nM T64682 D0D6DH 10125830 IC50 > 50000 nM T64682 D0F3FC 25022668 IC50 = 13 nM T64682 D0J3LR 11634725 Ki > 10000 nM T64682 D0Q3NG 11715520 Ki > 9400 nM T64682 D0S7IE 11658882 Ki > 9400 nM T72491 D0A7MY 637568 EC50 = 5110 nM T72491 C2UAY1 10455 IC50 > 100000 nM T72491 CKT98D 206035 IC50 > 100000 nM T72491 C9LYF4 286388 IC50 > 25000 nM T72491 CHCF90 665797 IC50 = 3000 nM T72491 CUHT06 899644 IC50 > 25000 nM T72491 CR5D2O 1070170 IC50 > 100000 nM T72491 COY71L 1073725 IC50 = 1800 nM T72491 CAP82W 1103353 IC50 > 25000 nM T72491 CG6UE9 1358452 IC50 = 2800 nM T72491 C60USN 1367926 IC50 > 25000 nM T72491 C9BPG3 1381629 IC50 = 890 nM T72491 CI5C4F 2133805 EC50 = 2900 nM T72491 CL8I0S 2772227 IC50 > 100000 nM T72491 C45EWL 3307826 EC50 > 100000 nM T72491 CXP4D9 6875758 EC50 = 9800 nM T72491 CCDG85 7514662 EC50 = 1120 nM T72491 C7GXT1 8814789 EC50 = 1060 nM T72491 CE2H5T 8814806 EC50 = 1770 nM T72491 CAH31D 8827213 EC50 = 1460 nM T72491 C4PX7O 9815648 IC50 > 100000 nM T72491 CHEX59 10329524 IC50 > 100000 nM T72491 CU79FN 16328219 EC50 = 1460 nM T72491 C1KP4N 40482356 IC50 = 2300 nM T72491 C8FD7E 40482358 EC50 > 100000 nM T72491 CZQ64N 44787480 IC50 > 25000 nM T72491 C8Z3UM 45040448 IC50 > 100000 nM T72491 C3EW7A 50744391 EC50 = 118000 nM T72491 C7PZ9N 56840728 EC50 = 2300 nM T72491 CYVK20 60149024 IC50 = 50118.72 nM T72491 C5HC3B 71681615 IC50 = 22 nM T72491 C3FVN4 71772353 IC50 > 100000 nM T72491 CK3SA1 71812184 EC50 = 1360 nM T72491 C6KD9Z 72189661 EC50 = 2420 nM T72491 C8IB1P 72189966 EC50 = 1630 nM T72491 C1LT8Q 72189968 EC50 = 2060 nM T72491 CS4QL7 72189970 EC50 = 2430 nM T72491 CAN4Z5 72771091 IC50 = 7400 nM T72491 CP7H8X 72771092 IC50 = 750 nM T72491 C38YIA 72771096 IC50 = 1100 nM T72491 C4O1IR 73330369 IC50 = 29 nM T72491 C82RVX 75202265 IC50 > 100000 nM T72491 CH9R1G 77461035 EC50 = 28.6 nM T72491 CBR20Z 91885637 IC50 = 63 nM T72491 CZ8YW7 96002439 EC50 = 5000 nM T72491 CXR0O8 106325804 IC50 > 100000 nM T72491 CXD39Z 118170767 EC50 = 12 nM T72491 C58FEG 118735935 IC50 = 750 nM T72491 CY3QN9 119057445 IC50 = 6200 nM T72491 C1U5AZ 122184660 IC50 = 980 nM T72491 CWY1V7 122184773 IC50 = 966 nM T72491 C1KQ4F 122184774 IC50 = 1666 nM T72491 CBS41H 122184775 IC50 = 10170 nM T72491 C60DTL 122184776 IC50 = 602 nM T72491 C2LR8K 122184777 IC50 = 18.1 nM T72491 C21HBC 122184778 IC50 = 54.3 nM T72491 CI2EZ4 122184779 IC50 = 42.3 nM T72491 CJ07IS 122184780 IC50 = 36.5 nM T72491 CF2MP3 122184781 IC50 = 14.4 nM T72491 CA2T7W 122184782 IC50 = 50.2 nM T72491 CP5NL4 122184783 IC50 = 979 nM T72491 C0OT6L 122184784 IC50 = 34.3 nM T72491 C1MG4H 122184785 IC50 = 179 nM T72491 C47JOU 122184786 IC50 = 47.4 nM T72491 CB9WT4 122184787 IC50 = 122 nM T72491 C1ISB2 122184788 IC50 = 66.1 nM T72491 CR4W6T 122184789 IC50 = 118 nM T72491 CHXM60 122184790 IC50 = 42.2 nM T72491 CL4WB3 122184791 IC50 = 1860 nM T72491 CP9N7W 122190547 EC50 = 5400 nM T72491 CKX08N 122190548 EC50 = 17100 nM T72491 CZL7X3 122190554 EC50 = 11500 nM T72491 CADN59 122190579 EC50 = 20600 nM T72491 C8FU3D 122190580 EC50 = 10000 nM T72491 C1B9FH 122190581 EC50 = 37800 nM T72491 CHS9C4 122190582 EC50 = 22600 nM T72491 C1IXV8 122190583 EC50 = 15000 nM T72491 CR48TK 122190584 EC50 = 11300 nM T72491 C1ID6T 122190585 EC50 = 15000 nM T72491 C96VNR 122190586 EC50 = 38500 nM T72491 C6UNI5 122190587 EC50 = 12700 nM T72491 CMCH49 122190589 EC50 = 8800 nM T72491 C4VK5C 122190590 EC50 = 24500 nM T72491 COC0V8 122190591 EC50 = 7100 nM T72491 C9G2JO 122194678 IC50 = 630 nM T72491 C3TG7O 122194679 IC50 > 25000 nM T72491 C4G5CV 122194680 IC50 > 25000 nM T72491 CPN19J 122194681 IC50 = 1100 nM T72491 CKT2A0 122194682 IC50 = 190 nM T72491 C4U7RN 122194683 IC50 = 660 nM T72491 CE45IP 122194684 IC50 > 25000 nM T72491 C2P8GB 122194685 IC50 > 25000 nM T72491 CA06HT 122194686 IC50 > 25000 nM T72491 CEI45M 122194687 IC50 > 25000 nM T72491 CNOL81 122194688 IC50 > 25000 nM T72491 CQ7NK0 122194689 IC50 > 25000 nM T72491 C9B5FT 122194690 IC50 > 25000 nM T72491 C5D3PT 122194808 IC50 > 25000 nM T72491 CJ28CN 122194809 IC50 = 410 nM T72491 C4KPW8 122194810 IC50 = 85 nM T72491 CLX1H2 122194811 IC50 > 25000 nM T72491 CB7DW0 122194812 IC50 > 25000 nM T72491 C5WZ9F 122194813 IC50 > 25000 nM T72491 CCVQ94 122194814 IC50 > 25000 nM T72491 CT0Q6I 122194815 IC50 = 5500 nM T72491 CGPU04 122194816 IC50 > 25000 nM T72491 C2RUM6 122194817 IC50 > 25000 nM T72491 C6H8SZ 126754132 IC50 < 10 nM T72491 CVL17P 134135178 IC50 = 320 nM T72491 C8IN5B 134139769 IC50 = 875 nM T72491 CLAP94 134141598 IC50 = 200 nM T72491 C9KCA0 134141909 IC50 = 230 nM T72491 CE8SA7 134145193 IC50 = 720 nM T72491 CT62RW 134148665 IC50 = 1300 nM T72491 CSW15J 134150874 IC50 = 634 nM T72491 C28GDW 134152173 IC50 = 3200 nM T72491 CU75YM 134155904 IC50 = 150 nM T72491 C0AG9Z 134813907 IC50 = 60 nM T72491 C85BCI 145951631 IC50 = 1100 nM T72491 CWKC32 145951903 IC50 > 25000 nM T72491 CJPS35 145952403 IC50 > 25000 nM T72491 C4XK3E 145952882 IC50 > 25000 nM T72491 C9N2PW 145952907 IC50 = 101 nM T72491 CIR3D0 145954661 IC50 = 1300 nM T72491 CR67LU 145955145 IC50 = 69700 nM T72491 CW3F9D 145956525 IC50 > 25000 nM T72491 C6UI5X 145956930 IC50 > 25000 nM T72491 CLG56Z 145957104 IC50 > 25000 nM T72491 C0T7QR 145971211 IC50 > 25000 nM T72491 CXLJ15 145973160 IC50 > 25000 nM T72491 CHO10Y 145974303 IC50 > 100000 nM T72491 C5OL0F 145975241 EC50 = 79 nM T72491 CD6L1Q 145979081 IC50 > 100000 nM T72491 CY6PF7 146680922 IC50 = 15.8 nM T72491 CJG46A 155510853 IC50 = 63095.73 nM T72491 C9VYG6 155511125 IC50 > 100000 nM T72491 CUY3M5 155511349 IC50 > 100000 nM T72491 CR01LK 155513180 IC50 = 50118.72 nM T72491 C7ON3W 155513257 IC50 = 19952.62 nM T72491 CK0R4I 155514102 IC50 > 100000 nM T72491 CJ3WP0 155514543 EC50 = 1390 nM T72491 CO9RY3 155515282 IC50 = 50118.72 nM T72491 CUT94K 155515491 EC50 = 970 nM T72491 CTJ97K 155516643 IC50 > 100000 nM T72491 CT28RK 155516991 IC50 = 39810.72 nM T72491 CC9K7R 155517070 IC50 = 50118.72 nM T72491 CYD95J 155517097 IC50 = 39810.72 nM T72491 CP68KM 155517263 IC50 = 50118.72 nM T72491 CB9MT8 155519311 IC50 = 15848.93 nM T72491 C68RTM 155519428 EC50 = 1360 nM T72491 CE6S0K 155519779 IC50 = 6309.57 nM T72491 C9TFN3 155520145 IC50 = 50118.72 nM T72491 C7PO4L 155520368 EC50 = 1910 nM T72491 CYX39S 155520897 EC50 = 1100 nM T72491 CUWL37 155521263 EC50 = 990 nM T72491 CA8IS0 155521928 IC50 = 19952.62 nM T72491 CL65ZK 155524194 IC50 > 100000 nM T72491 CS0WI3 155525300 IC50 = 2600 nM T72491 C73KQP 155525472 IC50 = 39810.72 nM T72491 C3MDZ4 155525522 IC50 > 100000 nM T72491 C4BAY9 155526259 IC50 > 100000 nM T72491 C8JU0Y 155526260 IC50 > 100000 nM T72491 C5RPQ3 155526688 IC50 > 100000 nM T72491 CJX51W 155527016 IC50 > 100000 nM T72491 C90REN 155527528 EC50 = 630 nM T72491 CEP71W 155528033 IC50 = 5011.87 nM T72491 CWI4Q5 155528195 IC50 = 50118.72 nM T72491 CCE2M5 155528362 IC50 > 100000 nM T72491 CS3QI5 155528453 EC50 = 3330 nM T72491 CFO37K 155528822 IC50 = 15848.93 nM T72491 C7L6CB 155529157 IC50 = 12589.25 nM T72491 C38UVP 155529704 IC50 = 12589.25 nM T72491 CKGA51 155530132 IC50 > 100000 nM T72491 C1ZTY3 155530152 IC50 = 63095.73 nM T72491 CEJQ10 155530334 IC50 = 3981.07 nM T72491 CQ4OC5 155531518 IC50 > 100000 nM T72491 CD5B4Z 155531917 IC50 > 100000 nM T72491 CCZ13G 155532065 IC50 = 50118.72 nM T72491 CU1A8Y 155532391 IC50 > 100000 nM T72491 C23ISL 155533277 EC50 = 1230 nM T72491 C7Q8UV 155533600 EC50 = 1540 nM T72491 CPH14B 155533997 IC50 > 50000 nM T72491 C2ZX3Y 155534140 EC50 = 2580 nM T72491 CWQ8P2 155534356 EC50 > 5000 nM T72491 C3K4EL 155535225 IC50 = 5011.87 nM T72491 C0Y9OK 155536020 IC50 = 39810.72 nM T72491 CF36VE 155536250 IC50 = 31622.78 nM T72491 COZC62 155536474 IC50 = 15848.93 nM T72491 CC64FE 155536577 IC50 = 50118.72 nM T72491 CO6ER7 155537046 IC50 = 25118.86 nM T72491 CW7AK4 155537439 IC50 = 15848.93 nM T72491 CK62ID 155537869 IC50 > 100000 nM T72491 C3WE9N 155538368 IC50 = 31622.78 nM T72491 C2RS7E 155539746 IC50 = 609 nM T72491 C75KYA 155540072 IC50 = 19952.62 nM T72491 C6PTE5 155540447 IC50 = 10000 nM T72491 CF0RT5 155540699 IC50 > 100000 nM T72491 CPFC16 155540797 IC50 = 63095.73 nM T72491 C67XKR 155541172 IC50 = 50118.72 nM T72491 C1L0WK 155541675 IC50 > 100000 nM T72491 C43NZV 155542200 IC50 = 10000 nM T72491 CQ8PW0 155542328 IC50 > 100000 nM T72491 CF2P7M 155542638 IC50 > 100000 nM T72491 C4MOF9 155543478 IC50 > 100000 nM T72491 CX8YP9 155543849 EC50 > 5000 nM T72491 C4G6RN 155544017 EC50 > 1000 nM T72491 C2M7EI 155544159 IC50 = 25118.86 nM T72491 C6JOP4 155545387 IC50 = 5011.87 nM T72491 C7UD2J 155546696 IC50 = 50118.72 nM T72491 CZ0I1S 155547074 IC50 > 100000 nM T72491 CQBT74 155547935 IC50 = 19952.62 nM T72491 CO7G5S 155548430 IC50 > 100000 nM T72491 C5XD8R 155548655 IC50 > 100000 nM T72491 C1V5OY 155548738 EC50 = 5520 nM T72491 CEPW05 155549226 IC50 = 100000 nM T72491 CT20GV 155549977 IC50 = 10000 nM T72491 CV4PU6 155550024 IC50 > 50000 nM T72491 CQ1TK8 155550838 EC50 = 1720 nM T72491 C5L8JE 155552136 IC50 > 100000 nM T72491 C9P1KN 155552525 IC50 > 50000 nM T72491 CDK9G7 155553288 IC50 = 2511.89 nM T72491 CH4G2N 155553767 IC50 > 100000 nM T72491 C8YIK6 155553920 IC50 = 25118.86 nM T72491 CNS6W1 155554404 EC50 = 1800 nM T72491 CBQ1U7 155554694 EC50 = 6970 nM T72491 CX83BF 155555686 IC50 = 39810.72 nM T72491 C6WPD1 155555697 IC50 = 50118.72 nM T72491 C0BPZ3 155555710 IC50 = 7943.28 nM T72491 C93OHG 155556364 IC50 = 31622.78 nM T72491 C8BQE6 155556461 IC50 = 15848.93 nM T72491 CQS7P0 155557407 IC50 = 39810.72 nM T72491 CB8Q5Y 155557794 IC50 = 12589.25 nM T72491 CL9F3S 155557868 IC50 = 25118.86 nM T72491 CRL16T 155558461 IC50 = 39810.72 nM T72491 C9XCN2 155558691 IC50 = 31622.78 nM T72491 C1C0ZO 155560119 EC50 = 2840 nM T72491 C24WDN 155560460 IC50 > 100000 nM T72491 CP2H0X 155560853 IC50 > 100000 nM T72491 CB63KG 155561425 IC50 > 100000 nM T72491 CEY87B 155562396 IC50 > 50000 nM T72491 CIJ0H9 155562696 IC50 > 100000 nM T72491 CB6NP3 155563580 IC50 = 31622.78 nM T72491 C13OYN 155563808 IC50 = 31622.78 nM T72491 CP61RM 155564286 IC50 = 31622.78 nM T72491 CA1K9B 155564526 IC50 = 7943.28 nM T72491 C4AL7M 155564597 IC50 > 100000 nM T72491 C85CMZ 155564705 IC50 = 25118.86 nM T72491 C1GUE5 155564896 EC50 = 2300 nM T72491 C6O4NA 155566445 IC50 = 25118.86 nM T72491 CF32ZO 155566614 IC50 > 100000 nM T72491 CC1H8N 155569160 IC50 > 50000 nM T72491 C5P6OE 155569644 IC50 > 100000 nM T72491 D0X4IO 5350 EC50 = 870 nM T06182 CB59HM 11570626 IC50 = 12800 nM T06182 CPLU74 60170970 IC50 = 2600 nM T06182 CX19CT 60170971 IC50 = 1700 nM T06182 CA0EO3 60171059 IC50 = 2600 nM T06182 CT4Z1R 127034614 IC50 = 53 nM T06182 CU12JI 127035881 IC50 = 36 nM T71192 D00QET 5281040 IC50 = 0.78 nM T71192 D05DVP 5717 IC50 = 14 nM T71192 D08QIP 4887 IC50 = 0.8 nM T71192 D00MHP 128355 IC50 = 23 nM T71192 D0U5YM 46830962 IC50 = 1.7 nM T71192 D09DIG 57109 IC50 = 4000 nM T71192 C9T3FB 105007 IC50 = 4000 nM T71192 C8RBI4 159289 IC50 = 2200 nM T71192 CA5OL4 5311184 IC50 = 23 nM T71192 C0EM5S 6509849 IC50 = 8 nM T71192 C0ZG5O 9804436 IC50 = 2.7 nM T71192 CY9MA1 9809348 IC50 = 0.55 nM T71192 C50ESJ 9829145 IC50 = 0.19 nM T71192 C34ABL 9829999 IC50 = 1.91 nM T71192 CG6ZK5 9890153 IC50 = 11 nM T71192 CK63UJ 10053523 IC50 = 44 nM T71192 CFN61X 10074704 IC50 = 3.4 nM T71192 C7XC2W 10324292 IC50 = 38 nM T71192 CUC5L8 10436360 IC50 = 4000 nM T71192 CLH69R 10502162 IC50 = 270 nM T71192 COK3Q2 10532372 IC50 = 63 nM T71192 CD3TW2 10553494 IC50 = 31 nM T71192 C45JMU 10574284 IC50 = 17 nM T71192 C0K8XO 10576732 IC50 = 300 nM T71192 CU8YK9 10597232 IC50 = 346 nM T71192 C6AX4M 10597634 IC50 = 31 nM T71192 C3WXD1 10598159 IC50 = 408 nM T71192 C0XVO8 10600630 IC50 = 45 nM T71192 CL0XQ8 10646529 IC50 = 105 nM T71192 C8T3BA 10647443 IC50 = 6.6 nM T71192 CLG24O 10649046 IC50 = 207 nM T71192 CP0V1A 10649109 IC50 = 500 nM T71192 C7U1HV 10651746 IC50 = 382 nM T71192 C9MN5W 10717271 IC50 = 609 nM T71192 CZP82W 10764001 IC50 = 143 nM T71192 CLAW26 10764782 IC50 = 1100 nM T71192 CU3M7I 10765224 IC50 = 13 nM T71192 C18NCQ 10766366 IC50 = 104 nM T71192 CO1SI2 10767627 IC50 = 17 nM T71192 CAM73P 10787157 IC50 = 1700 nM T71192 CAIJ24 10790119 IC50 = 1700 nM T71192 CISP89 10792471 IC50 = 12 nM T71192 CJ50HX 10836131 IC50 = 450 nM T71192 CUQ3E2 10836133 IC50 = 415 nM T71192 C59QLA 10839186 IC50 = 101 nM T71192 CO8KI0 11191817 IC50 = 11 nM T71192 CS0J3E 11227280 IC50 = 22 nM T71192 CFMP93 11249398 IC50 = 58 nM T71192 CA5G8V 11261220 IC50 = 0.59 nM T71192 CGHR62 11284237 IC50 = 32 nM T71192 CC9VH6 11307317 IC50 = 120 nM T71192 CK9ST2 11353238 IC50 = 35 nM T71192 C91OUF 11387037 IC50 = 51 nM T71192 C3TL2O 11398475 IC50 = 17 nM T71192 CW8D7G 11398820 IC50 = 0.79 nM T71192 CC1S3B 11455387 IC50 = 24 nM T71192 CGX8F6 11596869 IC50 = 24.1 nM T71192 CNC9T1 11626955 IC50 = 112 nM T71192 C57MBJ 11690196 IC50 = 1430 nM T71192 C69TXN 11713438 IC50 = 1.5 nM T71192 C7O2VK 11796528 IC50 = 530 nM T71192 CWH9Q3 11853184 IC50 = 13 nM T71192 C2E4QJ 14325224 IC50 = 3.1 nM T71192 C5E3WA 14742716 Ki = 11 nM T71192 C1U4XR 15290701 IC50 = 8.49 nM T71192 C1EZ6I 15290705 IC50 = 1.16 nM T71192 C31YRP 15290709 IC50 = 0.76 nM T71192 CO9HI1 15291439 IC50 = 2.7 nM T71192 CJK59F 15291441 IC50 = 2.4 nM T71192 C2YWT5 15291446 IC50 = 0.5 nM T71192 CRC07E 15291450 IC50 = 190 nM T71192 C45JZF 23124563 IC50 = 1.4 nM T71192 CKGH56 23124623 IC50 = 1300 nM T71192 CROH42 23124629 IC50 = 12 nM T71192 C3HYZ8 23124664 IC50 = 70 nM T71192 CLW5A4 23124672 IC50 < 1 nM T71192 C1L5NF 23124680 IC50 = 70 nM T71192 CDCT78 23124707 IC50 = 82 nM T71192 C9NAV8 23124716 IC50 = 290 nM T71192 CE8S9N 23124741 IC50 = 3000 nM T71192 CXQ38G 23124775 IC50 = 130 nM T71192 CRW4V9 23663996 IC50 = 310 nM T71192 CWF50E 44319586 IC50 = 15.7 nM T71192 CC5IT1 44319587 IC50 = 2.01 nM T71192 C2LRG6 44319715 IC50 = 0.72 nM T71192 CVP1U9 44319716 IC50 = 6.42 nM T71192 CC40AI 44319717 IC50 = 0.65 nM T71192 C4U6ML 44319718 IC50 = 0.47 nM T71192 CNL60U 44319774 IC50 = 8.67 nM T71192 CC49QG 44319782 IC50 > 150 nM T71192 CQ8NH0 44319783 IC50 = 1.06 nM T71192 CM0Y3J 44319827 IC50 = 3.36 nM T71192 CRQP48 44319872 IC50 = 2.16 nM T71192 CC58WV 44319977 IC50 = 4.7 nM T71192 CT3Z7O 44319978 IC50 = 2.43 nM T71192 CC5T1W 44319992 IC50 = 1.63 nM T71192 CC46HF 44320021 IC50 = 1.05 nM T71192 C81BFE 44320022 IC50 = 0.38 nM T71192 C9NKG4 44322990 IC50 = 3.1 nM T71192 C8EKY0 44352103 IC50 = 8.4 nM T71192 CW2DK3 44352142 IC50 = 44 nM T71192 CM9KZ8 44352148 IC50 = 7.3 nM T71192 C64KME 44352154 IC50 = 9.2 nM T71192 CW70IG 44352186 IC50 = 9 nM T71192 CB27NK 44352282 IC50 = 13 nM T71192 C35PDK 44352288 IC50 = 21 nM T71192 C2LMA4 44352294 IC50 = 4.6 nM T71192 C3OJU2 44352326 IC50 = 7.3 nM T71192 CR68MH 44352397 IC50 = 86 nM T71192 CU7FT1 44352406 IC50 = 1.5 nM T71192 C49ILY 44352450 IC50 = 30 nM T71192 CQI2V7 44352452 IC50 = 3.8 nM T71192 CUM51E 44352484 IC50 = 38 nM T71192 CX9HR4 44360585 IC50 = 0.47 nM T71192 C1U4HZ 44360625 IC50 = 1.1 nM T71192 CDZ5V1 44360637 IC50 = 0.9 nM T71192 C0MH5O 44360640 IC50 = 2 nM T71192 C3F8DC 44360643 IC50 = 0.21 nM T71192 CB3PX8 44360644 IC50 = 2.9 nM T71192 CB21JX 44360674 IC50 = 0.34 nM T71192 CRHZ26 44360675 IC50 = 1.7 nM T71192 CLY2J8 44360752 IC50 = 4.9 nM T71192 C9WI8M 44360808 IC50 = 421 nM T71192 CO6UZ0 44360844 IC50 = 5 nM T71192 C9W7TQ 44360858 IC50 = 0.42 nM T71192 C2KH6D 44360895 IC50 = 25.2 nM T71192 CSB4R8 46830677 IC50 = 2.8 nM T71192 C9BHQ2 46830961 IC50 = 3.4 nM T71192 C9DXV5 46830963 IC50 = 7.4 nM T71192 C9BT3C 46834997 IC50 = 1.5 nM T71192 C3OD2Q 46835000 IC50 = 1.1 nM T71192 C4O3AD 46919026 EC50 = 480 nM T71192 C5OXF1 49863579 IC50 = 810 nM T71192 CUP2Y8 49863608 IC50 = 2100 nM T71192 CUF1T9 49863609 IC50 = 34000 nM T71192 COE89A 49863641 IC50 = 55000 nM T71192 CINV43 49863643 EC50 = 1400 nM T71192 CYAZ59 49863644 EC50 = 1300 nM T71192 CI94PA 49863685 EC50 = 3900 nM T71192 C1IKC0 49863766 IC50 = 15 nM T71192 C07RZF 49863809 IC50 = 36 nM T71192 CL68EN 49863872 IC50 = 168 nM T71192 C1B0NP 49863895 IC50 = 10500 nM T71192 CAU02Q 49863907 IC50 = 2 nM T71192 CI7PE4 49863921 IC50 = 4.1 nM T71192 CR42SZ 49863922 IC50 = 4 nM T71192 CCI1M9 49863923 IC50 = 5 nM T71192 COB69G 49863945 IC50 = 14 nM T71192 CXB41R 49863972 IC50 = 130 nM T71192 C4FGC6 54677430 IC50 = 9700 nM T71192 CW70SA 59599459 IC50 = 330 nM T71192 CF45DO 59599475 IC50 = 1500 nM T71192 C12XMG 59599515 IC50 = 132 nM T71192 CIB19F 59599538 IC50 = 346 nM T71192 CC8W5L 59599545 IC50 = 342 nM T71192 CJIV72 59599552 IC50 = 475 nM T71192 C3OAM1 59599555 IC50 = 390 nM T71192 C1MJ8Z 59599565 IC50 = 200 nM T71192 CF3TQ4 59599568 IC50 = 203 nM T71192 CV91KQ 59599576 IC50 = 73.6 nM T71192 C1VAB2 59599577 IC50 = 62.4 nM T71192 CD5T6R 59599580 IC50 = 144 nM T71192 CHX74C 59599616 IC50 = 484 nM T71192 CLGZ72 66739117 IC50 = 0.56 nM T71192 CJ7PE4 68695885 IC50 = 3.4 nM T71192 C2DCQ4 87131159 IC50 = 1.6 nM T71192 CC01GT 90871050 IC50 = 54 nM T71192 CX83VY 118716772 IC50 = 4600 nM T71192 CNYK86 118716773 IC50 = 840 nM T71192 C0B3PZ 118716774 IC50 = 13 nM T71192 C81NVL 118716775 IC50 = 150 nM T71192 CSTV67 118716776 IC50 = 300 nM T71192 CHM06D 118716777 IC50 = 44 nM T71192 C8OAM0 118728613 IC50 = 1900 nM T71192 C2E5LC 118729613 IC50 = 740 nM T71192 CHV59E 118729614 IC50 = 250 nM T71192 CI48HX 118729615 IC50 = 490 nM T71192 CU8GO5 122183681 IC50 = 3.1 nM T71192 C57LAY 122183682 IC50 = 1 nM T71192 CD2X9M 122183683 IC50 = 2.9 nM T71192 CBZT62 122183684 IC50 = 0.62 nM T71192 CXY1J3 122183685 IC50 = 4.1 nM T71192 C8JPS5 122183686 IC50 = 46 nM T71192 C9GY0M 122183687 IC50 = 2.4 nM T71192 C7LR4C 122183688 IC50 = 2.2 nM T71192 C3SBE6 122183689 IC50 = 0.8 nM T71192 CI83YC 122183690 IC50 = 1.1 nM T71192 C6SP3V 122183751 IC50 = 0.47 nM T71192 CIWZ15 122183752 IC50 = 0.32 nM T71192 CMV47L 122183753 IC50 = 0.22 nM T71192 C25ETG 122183754 IC50 = 12 nM T71192 CC91EO 122183755 IC50 = 10 nM T71192 CH4K5P 122183756 IC50 = 17 nM T71192 C3DML9 122183757 IC50 = 5.5 nM T71192 C0IMN8 122183758 IC50 = 0.79 nM T71192 C9YGC0 122183759 IC50 = 65 nM T71192 CA7P1R 122183760 IC50 = 25 nM T71192 CFD79M 122183761 IC50 = 56 nM T71192 CV9G8Y 122183762 IC50 = 16 nM T71192 C1GI5T 122183763 IC50 = 11 nM T71192 C8K9XA 122196341 IC50 > 1200 nM T71192 C1IQ0H 127043048 IC50 = 31000 nM T71192 C0WU9P 127043049 IC50 = 290 nM T71192 CA0V8Q 127043050 IC50 = 9 nM T71192 CUQL23 127043053 IC50 = 67 nM T71192 CW84IQ 127043233 IC50 = 120 nM T71192 CW5PI4 127043236 IC50 = 35 nM T71192 CFB30X 127043237 IC50 = 58 nM T71192 C1A0OU 127043241 IC50 = 17 nM T71192 COHV05 127043242 IC50 = 22 nM T71192 CM78QW 127043243 IC50 = 16 nM T71192 CU79CR 127043244 IC50 = 7.8 nM T71192 CYL20V 127043247 IC50 = 38 nM T71192 CXA12T 127043248 IC50 = 25 nM T71192 CSJF19 127043252 IC50 = 660 nM T71192 C3ULM6 127043253 IC50 > 100000 nM T71192 CT6Y3D 127043406 IC50 > 100000 nM T71192 CF42NI 127043407 IC50 > 100000 nM T71192 CP5Q0G 127043408 IC50 > 100000 nM T71192 C39QTB 127043409 IC50 > 100000 nM T71192 C6CY1T 127043410 IC50 > 100000 nM T71192 C0X9QH 127043411 IC50 > 100000 nM T71192 CD89CS 127043617 IC50 = 12 nM T71192 CM84GW 127043618 IC50 = 5.9 nM T71192 CP0D1Z 127044872 IC50 > 100000 nM T71192 C9PS6W 127045334 IC50 > 100000 nM T71192 CS2T5L 127045343 IC50 > 100000 nM T71192 CWVP43 135430849 IC50 = 14 nM T71192 C2TK8Q 136127005 IC50 = 527 nM T71192 D03YBH 5280878 Ki = 0.29 nM T71192 D05CNT 5311015 IC50 = 440 nM T71192 D06AYN 10438479 IC50 > 10000 nM T71192 D09JQU 53394034 IC50 > 2500 nM T71192 D0G7OZ 60842 Ki = 10 nM T73557 D0D1SG 5755 EC50 = 32 nM T73557 CR68MZ 6323453 Ki = 850 nM T73557 CYI7T4 9802231 EC50 = 53.7 nM T73557 C59VXD 10386752 EC50 = 14.2 nM T73557 CFVP19 10428095 EC50 = 66 nM T73557 CVQS04 10454813 EC50 = 37.7 nM T73557 CW6P7A 11244720 EC50 = 181.6 nM T73557 CXG0C2 11269006 EC50 = 66 nM T73557 C4SC0W 11281576 EC50 = 129.2 nM T73557 C2WVO7 13877991 Ki = 75000 nM T92640 C4Z7TA 128167 Ki = 407 nM T92640 CD2K9I 219925 IC50 > 7300 nM T92640 CNX1I9 744590 Ki = 50 nM T92640 C2MU3S 753410 Ki = 311 nM T92640 CYQ7L5 1365686 Ki = 48 nM T92640 C4TGR0 2260227 Ki = 13470 nM T92640 CN8XM2 5311263 EC50 = 17 nM T92640 CWIH09 5311306 Ki = 137 nM T92640 CAX9U1 5473680 EC50 > 12300 nM T92640 CLS96Y 6419701 EC50 = 70.79 nM T92640 C9R7UG 6610239 EC50 = 1850 nM T92640 CA78VE 9958483 IC50 = 89 nM T92640 C9EQ7R 9960370 IC50 > 10000 nM T92640 C8IGL1 10136738 EC50 = 221 nM T92640 COZF72 10322404 EC50 = 14.7 nM T92640 CE1Y9O 10393842 Ki = 18 nM T92640 C9TW5S 10432332 EC50 = 318 nM T92640 CLJ0N4 11101949 Ki = 221 nM T92640 C78IDM 11167018 IC50 = 140 nM T92640 CK12CR 11236547 IC50 = 130 nM T92640 C3FJ8O 11271067 IC50 = 23 nM T92640 CTHF04 11305821 IC50 = 170 nM T92640 CF4SM5 11316893 IC50 = 130 nM T92640 CRZT82 11317548 IC50 = 0.16 nM T92640 CNU29D 11340921 IC50 = 430 nM T92640 CW5Z0B 11351723 IC50 = 61 nM T92640 C3JYZ0 11374611 IC50 = 220 nM T92640 C2MD0Q 11409276 IC50 = 280 nM T92640 CQLP42 11473989 EC50 = 193 nM T92640 CRCF96 11512311 IC50 > 10000 nM T92640 CFHV74 11568387 Ki = 360 nM T92640 C2JDN7 11592067 IC50 > 10000 nM T92640 CIZW04 11599847 Ki = 358 nM T92640 C0CBY2 11625765 EC50 = 695 nM T92640 C7QRT8 11648176 EC50 = 8.318 nM T92640 CK7O0X 11849496 Ki = 314 nM T92640 CF5O3H 16016731 IC50 = 800000 nM T92640 CR79CQ 16043259 Ki = 403 nM T92640 CGW71D 23079111 IC50 = 390 nM T92640 C0HDK8 23080067 IC50 = 1700 nM T92640 C70ONJ 23725184 Ki = 143 nM T92640 C1F9GI 24882686 IC50 > 50000 nM T92640 CR2M4K 44325214 IC50 = 7970 nM T92640 C6KE2Z 44325235 IC50 = 9030 nM T92640 C15FHI 44325304 IC50 > 10000 nM T92640 CW3XH1 44325312 IC50 = 4250 nM T92640 CI2YX1 44325339 IC50 > 10000 nM T92640 C9ZNP8 44325351 IC50 > 10000 nM T92640 CT82OZ 44325364 IC50 > 10000 nM T92640 CS0A5D 44325365 IC50 > 10000 nM T92640 COS7A5 44325366 IC50 > 10000 nM T92640 CT0RI4 44325370 IC50 > 10000 nM T92640 C16ENI 44325390 IC50 > 10000 nM T92640 CL6Q4T 44325391 Ki = 34 nM T92640 C8O6ZB 44325400 IC50 > 10000 nM T92640 CE1QC6 44325401 Ki = 134 nM T92640 C19LDV 44325402 IC50 > 10000 nM T92640 CG5N0T 44325416 IC50 > 10000 nM T92640 CD4AI9 44325421 IC50 > 10000 nM T92640 CDQ8P0 44325422 IC50 > 10000 nM T92640 CJI36T 44325680 IC50 > 10000 nM T92640 C2VWE0 44325681 Ki = 73 nM T92640 CMEB29 44325682 Ki = 156 nM T92640 C4F8UE 44343851 EC50 = 318 nM T92640 CD1SX3 44343866 EC50 = 40 nM T92640 CK0NG4 44343867 EC50 > 5000 nM T92640 C5J4BE 44343880 EC50 > 5000 nM T92640 CS7BJ1 44344023 EC50 = 1950 nM T92640 CV86RF 44368508 EC50 = 23.99 nM T92640 CD6ZL8 44392725 IC50 = 962 nM T92640 CV80NT 44392726 IC50 > 10000 nM T92640 CSQ0E4 44392727 IC50 > 10000 nM T92640 C0U3XC 44392738 IC50 > 10000 nM T92640 CHA7T6 44392762 IC50 = 4500 nM T92640 CP8S6X 44392769 IC50 = 735 nM T92640 CTKZ61 44392778 IC50 > 10000 nM T92640 CNVU84 44392779 IC50 = 2840 nM T92640 CXL4U0 44392780 IC50 > 10000 nM T92640 CUH71K 44392791 IC50 = 6250 nM T92640 C4Y8HZ 44392792 Ki = 26 nM T92640 CTNU76 44392793 Ki = 19 nM T92640 CM3RG9 44392794 Ki = 64 nM T92640 C1Y8ME 44392795 Ki = 35 nM T92640 CCOF81 44392796 Ki = 28 nM T92640 CKF5A4 44392797 IC50 = 3690 nM T92640 CGPA21 44392798 IC50 = 1430 nM T92640 CUR57A 44392834 IC50 > 10000 nM T92640 CR17IB 44392835 IC50 > 10000 nM T92640 CBR7Y6 44392836 IC50 > 10000 nM T92640 C5LAU4 44407386 Ki = 152 nM T92640 C9P3SU 44407394 Ki = 486 nM T92640 C9E2RP 44407397 EC50 = 3260 nM T92640 CWN45J 44407485 Ki = 2850 nM T92640 C8OB1A 44414925 Ki = 60.7 nM T92640 C3SX2V 44414935 EC50 > 1940 nM T92640 C1UB5L 44441080 IC50 = 260 nM T92640 CV7TA6 44441086 IC50 > 40000 nM T92640 C4TRN7 44441093 IC50 = 200 nM T92640 C25HPU 44441096 IC50 = 370 nM T92640 C29TWV 44454059 IC50 > 50000 nM T92640 CO7L3S 44454369 IC50 = 50 nM T92640 C85ANH 46213949 IC50 = 150 nM T92640 CET63X 46223906 EC50 = 16.5 nM T92640 C8CK4M 46240292 IC50 = 17 nM T92640 CO3DB1 56943915 IC50 = 6.6 nM T92640 CRP98X 58902982 IC50 = 61 nM T92640 CFSU32 59520112 IC50 = 2490 nM T92640 CNM5Y7 66553162 IC50 = 20 nM T92640 CA0D4Z 66773644 IC50 = 260 nM T92640 C5LE7W 66773650 IC50 = 260 nM T92640 C8JY6F 66773671 IC50 = 680 nM T92640 C6Y8QC 66773977 IC50 = 210 nM T92640 C6UY3N 66774140 IC50 > 1000 nM T92640 CLGK10 66774229 IC50 = 3300 nM T92640 CZQR78 66774300 IC50 = 1300 nM T92640 CPZR04 66774362 IC50 = 3700 nM T92640 C63XKM 66774424 IC50 = 230 nM T92640 C9GQ2D 66774612 IC50 = 100 nM T92640 C8I1QZ 66774667 IC50 = 190 nM T92640 C4ABK5 66774701 IC50 = 220 nM T92640 CW2O5R 66774777 IC50 = 3.5 nM T92640 C1PVS0 66774778 IC50 = 15 nM T92640 CJ6GD7 66774888 IC50 = 71 nM T92640 C6O5UJ 66774954 IC50 > 10000 nM T92640 CYJ67P 66774976 IC50 = 5500 nM T92640 CKL76D 66775043 IC50 = 160 nM T92640 CE6W9S 66775139 IC50 > 1000 nM T92640 CMZ35C 66775150 IC50 = 6600 nM T92640 CIN6V5 66775156 IC50 = 4400 nM T92640 CJUE12 66775301 IC50 = 5.9 nM T92640 CL4IE5 66775340 IC50 = 460 nM T92640 C2TSL8 66775429 IC50 = 12100 nM T92640 C9IVD3 66775552 IC50 = 130 nM T92640 CSJO90 66861497 IC50 = 34 nM T92640 CY1SR0 66861759 IC50 = 22 nM T92640 C7J4WG 66861761 IC50 = 40 nM T92640 CJ39PD 66861902 IC50 = 38 nM T92640 CREL14 66862202 IC50 = 29 nM T92640 C9KW8A 66862428 IC50 = 520 nM T92640 C02ZAJ 66862629 IC50 = 30 nM T92640 CA59XL 66862638 IC50 = 180 nM T92640 CBZ4X0 66862841 IC50 = 32 nM T92640 CZ52TI 66862949 IC50 = 45 nM T92640 CV10SQ 66863259 IC50 = 13 nM T92640 C5C4FO 70819309 IC50 = 106 nM T92640 C9NYD7 70819486 IC50 = 3590 nM T92640 C7GFM8 70819507 IC50 = 35 nM T92640 CN13BI 70856266 IC50 = 18 nM T92640 C19LCA 71264582 IC50 < 50 nM T92640 C4IVB2 71265339 IC50 = 25.2 nM T92640 CD7L0B 71267051 IC50 = 36 nM T92640 CO8X7S 71450321 IC50 = 398 nM T92640 CO06XW 71450322 IC50 = 32 nM T92640 CR6LV5 71452129 IC50 = 19 nM T92640 C8BJ1R 71452130 IC50 = 24 nM T92640 CLZI05 71452131 IC50 = 57 nM T92640 CMTN57 71453959 IC50 = 112 nM T92640 CET67P 71453960 IC50 = 48 nM T92640 CJ4ZR7 71453961 IC50 > 30000 nM T92640 C2YZP4 71455702 IC50 = 174 nM T92640 C43TXF 71455703 IC50 = 20 nM T92640 C80YTO 71455704 IC50 = 2650 nM T92640 CC86ZE 71457478 IC50 = 161 nM T92640 CN9YG6 71457479 IC50 = 70 nM T92640 CQMU34 71457480 IC50 = 17 nM T92640 CZH0Q5 71457481 IC50 = 24 nM T92640 CI4T3M 71457482 IC50 = 58 nM T92640 C2YO9B 71457483 IC50 = 17500 nM T92640 C38EKM 71459352 IC50 = 176 nM T92640 CF63KB 71459353 IC50 = 42 nM T92640 CPT4O8 71461120 IC50 = 34.5 nM T92640 CZW96E 71461121 IC50 = 985 nM T92640 CG0ZL8 71461122 IC50 > 30000 nM T92640 C2MPI8 71461123 IC50 > 30000 nM T92640 C4NU2T 71461124 IC50 = 3970 nM T92640 CID7N8 71461125 IC50 > 30000 nM T92640 C4QTR2 71462858 IC50 = 41 nM T92640 CV1L8R 71462859 IC50 = 38 nM T92640 C69ZER 71462861 IC50 = 217 nM T92640 CBE42D 71462862 IC50 = 23 nM T92640 C06NYA 71462863 IC50 = 644 nM T92640 C57TYK 71569053 EC50 = 26 nM T92640 CSN3I7 71569056 EC50 = 12.2 nM T92640 CPT5S2 71718248 EC50 = 11.1 nM T92640 CKC4U7 71719457 EC50 = 30.9 nM T92640 C5P1CQ 71720690 EC50 = 10.1 nM T92640 CZYL51 73332314 IC50 = 79 nM T92640 CEZ5X6 73335984 IC50 = 586 nM T92640 C5BIA4 73335985 IC50 = 2940 nM T92640 CKPL89 73335987 IC50 = 825 nM T92640 CXEV94 73336082 IC50 = 74 nM T92640 C71ZPR 73336083 IC50 = 3358 nM T92640 CJIF23 73336084 IC50 = 805 nM T92640 CZ5HU4 73336085 IC50 = 510 nM T92640 CNP98L 73336174 IC50 = 111 nM T92640 CL3Y8J 89484779 IC50 > 800 nM T92640 CQ3PK4 90308914 IC50 > 800 nM T92640 C89FXZ 90309040 IC50 > 800 nM T92640 CYSQ05 90309100 IC50 > 800 nM T92640 CY3ZT1 90309524 IC50 > 800 nM T92640 CQ6B3X 90665720 Ki = 84 nM T92640 CNI96W 118728428 IC50 > 25000 nM T92640 C3O6KB 118728429 IC50 > 25000 nM T92640 C4U3DG 118728430 IC50 > 800 nM T92640 C8U0GE 118728431 IC50 > 800 nM T92640 C72NCP 118728432 IC50 > 25000 nM T92640 C2YHT8 118728433 IC50 > 25000 nM T92640 C4M3YA 118728434 IC50 > 25000 nM T92640 CG65XZ 122191108 Ki = 170 nM T92640 CKL42I 122191542 EC50 = 40 nM T92640 CQ3W8I 122191543 EC50 = 790 nM T92640 CWQ8Y3 122191544 IC50 = 1500 nM T92640 CO5Y0B 122191545 IC50 = 130 nM T92640 CP0SK1 132191124 IC50 = 6000 nM T92640 CS7XL2 132191134 IC50 = 18000 nM T92640 CXI92L 132191135 IC50 = 14000 nM T92640 CW2O1F 134145238 IC50 = 140 nM T92640 C6GTI5 134148024 IC50 = 42 nM T92640 CVOZ93 134153933 IC50 > 1000 nM T92640 CBH75C 134156371 IC50 = 100 nM T92640 C9QMB5 134156710 IC50 = 140 nM T92640 CZE6V7 140083418 IC50 = 120 nM T92640 C07OQK 142610742 IC50 = 4 nM T92640 C89NRQ 150134920 IC50 = 27 nM T92640 CH13WN 150336102 IC50 = 620 nM T92640 CU0E6Q 152069844 IC50 = 9 nM T92640 CYKS78 155153661 IC50 = 227 nM T92640 C1ADN8 155153676 IC50 = 5 nM T92640 D02LXI 10367662 IC50 = 160 nM T92640 D02RYR 11447695 IC50 > 10000 nM T92640 D03HLU 11276402 IC50 > 10000 nM T92640 D04BLL 11312382 Ki = 457 nM T92640 D04CJG 82327 Ki = 1082 nM T92640 D05TVG 23682233 Ki = 170 nM T92640 D07WLV 11219269 IC50 > 10000 nM T92640 D07YUV 11197104 Ki = 1146 nM T92640 D0BP3E 11393306 Ki = 788 nM T92640 D0G6XT 10051843 Ki = 4300 nM T92640 D0GH9J 44407389 Ki = 139 nM T92640 D0P7GR 78401 IC50 ~ 10000 nM T92640 D0PI4H 10282223 IC50 = 2490 nM T92640 D0R8LB 44343825 EC50 = 197 nM T92640 D0S6CW 44392752 IC50 = 992 nM T92640 D0X0OP 56947064 EC50 = 571 nM T92640 D0X0UR 5497152 EC50 = 80 nM T92640 D0XJ9P 75816 Ki = 1354 nM T76024 D07XHO 4413 IC50 = 29 nM T76024 D01IBO 9822205 IC50 = 1.6 nM T76024 C7BU1L 2138 Ki = 12589.25 nM T76024 COHM79 117475 Ki = 100000000 nM T76024 CD14RN 197789 Ki = 251188.64 nM T76024 C2HTG4 229074 Ki > 100000000 nM T76024 CU4G3Y 309369 Ki = 15848.93 nM T76024 C2J3VS 576480 Ki = 1584893.19 nM T76024 C40DHV 3016780 Ki > 100000000 nM T76024 CB58JC 3357702 Ki = 79432.82 nM T76024 CZ9ST3 3564407 Ki = 251188.64 nM T76024 C7ZTI9 3676069 Ki = 6309573.44 nM T76024 C8EK6S 4620241 Ki = 100000 nM T76024 C9SJZ7 5048318 Ki > 100000000 nM T76024 CV95FQ 5108695 Ki = 158489.32 nM T76024 CG7BH6 5221300 Ki = 125892.54 nM T76024 CKN89B 9822176 Ki = 470 nM T76024 CFR6T1 9822409 Ki = 30 nM T76024 C73DNO 9908936 Ki = 3000 nM T76024 C8C6UI 9929077 Ki = 436 nM T76024 C1LCO8 10335742 Ki = 3000 nM T76024 C84THX 10424840 Ki = 6000 nM T76024 CPO7X4 11250283 Ki = 20 nM T76024 CIMH03 11852389 Ki = 11 nM T76024 CJL46R 12254250 Ki = 630957.34 nM T76024 C5PVL9 12456162 Ki = 501187.23 nM T76024 CA0Y5E 16219042 Ki = 31622.78 nM T76024 CW2LR9 18536775 Ki = 700 nM T76024 CH3FI0 18536798 Ki = 11000 nM T76024 CIM3R5 18536877 Ki = 850 nM T76024 C3FPX2 18536880 Ki = 420 nM T76024 C3GZT0 18536889 Ki = 560 nM T76024 CZL15E 18536922 Ki = 1000 nM T76024 CZON79 18536933 Ki > 20000 nM T76024 CBF3V5 18536936 Ki = 14400 nM T76024 CR0MI2 18537006 Ki = 870 nM T76024 CJ2DQ9 18537029 Ki = 960 nM T76024 C6CDS5 18537037 Ki = 900 nM T76024 CE38OR 18537047 Ki = 1020 nM T76024 CUL10T 18537184 Ki = 15400 nM T76024 CRJ81N 18537194 Ki = 1060 nM T76024 C2P7AX 18537198 Ki = 850 nM T76024 CVYU03 18537269 Ki = 750 nM T76024 CT6S1B 18537287 Ki = 860 nM T76024 CT9D4Y 18537290 Ki = 4700 nM T76024 C6PR7W 18537298 Ki = 490 nM T76024 CZO7I0 18537342 Ki = 520 nM T76024 CJH4D2 18537468 Ki = 640 nM T76024 CJ1S4P 18537474 Ki > 20000 nM T76024 C2QIV5 18672193 Ki = 30 nM T76024 C9JKF8 18672225 Ki = 60 nM T76024 C4I2LN 21057033 Ki = 64 nM T76024 CQ3LD7 21057057 Ki = 70 nM T76024 C1ZK9R 21057058 Ki = 30 nM T76024 C5F0JE 21057059 Ki = 400 nM T76024 C5QMH1 21057060 Ki = 1790 nM T76024 CY5WF9 21057067 Ki = 20 nM T76024 CFVT21 21057073 Ki = 460 nM T76024 CPS6N8 21057081 Ki = 150 nM T76024 C4AE1H 21057101 Ki = 210 nM T76024 CYL54R 21057103 Ki = 400 nM T76024 C9E6IC 21057104 Ki = 420 nM T76024 C6DHU7 21057134 Ki = 40 nM T76024 CO4BJ6 21057135 Ki = 30 nM T76024 CJR7Z6 21057138 Ki = 400 nM T76024 CGT93C 21057139 Ki = 310 nM T76024 CHVL05 21057140 Ki = 240 nM T76024 CT3B8D 21057141 Ki = 160 nM T76024 CUG5Z9 21057142 Ki = 170 nM T76024 CI81YV 21057144 Ki = 170 nM T76024 C7DQY9 21057146 Ki = 200 nM T76024 C6ARJ5 21057148 Ki = 330 nM T76024 CMG39P 21057150 Ki = 100 nM T76024 CL9TB2 21057156 Ki = 580 nM T76024 CEZ89C 21057157 Ki = 410 nM T76024 C5X4IQ 21057162 Ki = 260 nM T76024 CK58SP 21057183 Ki = 120 nM T76024 CBYC10 21057185 Ki = 14 nM T76024 C6UBT3 21886028 Ki = 1880 nM T76024 CIE0X3 21886048 Ki = 490 nM T76024 CO5T4N 21886122 Ki = 50 nM T76024 C9H0XG 21886127 Ki = 140 nM T76024 CHE12K 21886140 Ki = 40 nM T76024 CBO6E0 21886156 Ki = 42 nM T76024 CU3I1L 21886160 Ki = 100 nM T76024 C6I2OG 21886212 Ki = 360 nM T76024 C6M9YC 21886215 Ki = 400 nM T76024 CJ0GZ6 21886217 Ki = 120 nM T76024 CFPH59 21886223 Ki = 180 nM T76024 CIN7M8 21886237 Ki = 190 nM T76024 C0WYI1 21886261 Ki = 6 nM T76024 CPF90J 21886276 Ki = 250 nM T76024 C90RGC 21886301 Ki = 150 nM T76024 C4IJR3 21886316 Ki = 610 nM T76024 C13KGQ 21886365 Ki = 350 nM T76024 CZ15WT 21886367 Ki = 1850 nM T76024 CIR47A 21886371 Ki = 50 nM T76024 C5O9JL 21886763 Ki = 22 nM T76024 C54UVP 43165100 Ki = 10000000 nM T76024 C0B1XM 44278581 Ki = 450 nM T76024 CU81AY 44333788 Ki = 330 nM T76024 CTLH60 44333799 Ki = 190 nM T76024 CQSA02 44333829 Ki = 150 nM T76024 C4QT8G 44333831 Ki = 90 nM T76024 CEZV36 44333832 Ki = 530 nM T76024 C5M2LB 44333833 Ki = 70 nM T76024 CG4B1O 44333850 Ki = 1500 nM T76024 C7BE4R 44334067 Ki > 20000 nM T76024 C3T6LW 44334085 Ki > 28000 nM T76024 CDA6M3 44334096 Ki = 12500 nM T76024 CZ2G3P 44334110 Ki = 460 nM T76024 CFNA97 44334157 Ki = 3250 nM T76024 CHM61E 44410182 Ki = 2290 nM T76024 CB2PH8 44410205 Ki = 2240 nM T76024 C2R9ON 44410335 Ki = 2000 nM T76024 C72WFO 44410362 Ki = 380 nM T76024 CR17GB 44410372 Ki = 330 nM T76024 CPYM71 44447085 Ki = 40 nM T76024 CIKQ81 53345652 Ki > 130 nM T76024 CXWS90 53345968 Ki > 1000 nM T76024 CE5A7B 60162406 Ki > 100000 nM T76024 C30ZKJ 71561420 Ki > 35000 nM T76024 C78DJQ 71711730 IC50 < 10000 nM T76024 CG83WX 90655748 Ki > 100000000 nM T76024 CGL2B0 118725262 Ki = 199526.23 nM T76024 CDQ62V 137637214 Ki > 50000 nM T76024 C2K8JV 137639385 Ki > 50000 nM T76024 CNX46H 137654508 Ki > 50000 nM T76024 C8FST4 145985086 IC50 = 900 nM T76024 D0J1CC 11948634 Ki = 10 nM T76024 D0J2SM 296008 IC50 = 1250 nM T12817 C2Y6QS 50938552 IC50 > 10000 nM T12817 C9NYP4 51036677 IC50 > 10000 nM T12817 C4WRY3 51037112 IC50 > 10000 nM T12817 CRI28Z 51037948 IC50 > 10000 nM T12817 CY7BI2 118706214 IC50 > 10000 nM T12817 CHA4N2 136013680 IC50 > 10 nM T12817 C1YUD0 136219394 IC50 > 10 nM T12817 CIU8W3 136254389 IC50 > 10 nM T12817 D09HVH 135566652 IC50 > 10 nM T12817 D0H0AU 25195348 IC50 = 10400 nM T55260 CE4HM8 1032885 IC50 = 21000 nM T55260 C0KA3Q 3433760 IC50 = 31800 nM T55260 C9OV3N 6504357 IC50 = 42500 nM T55260 CNW5G7 9573924 IC50 = 20000 nM T55260 CKUQ62 10259546 IC50 = 230000 nM T55260 CJTN91 10345949 IC50 = 11000 nM T55260 CBUT60 10481524 IC50 = 3000 nM T55260 CF17EN 11840289 IC50 = 67800 nM T55260 CF43ME 44329918 IC50 = 400000 nM T55260 C58IRU 44329919 IC50 = 280000 nM T55260 COH27D 44329920 IC50 > 100000 nM T55260 C4V9NA 44330017 IC50 > 100000 nM T55260 C4Q1ST 44330324 IC50 = 45000 nM T55260 C83NEY 44330360 IC50 = 140000 nM T55260 C2FO7L 44330361 IC50 = 75000 nM T55260 D0O1BJ 445434 IC50 = 3 nM T50594 D05SBO 46220502 Ki < 10 nM T50594 D09DHY 6167 IC50 = 4300 nM T50594 D0K8KX 5280343 IC50 = 500 nM T50594 D0U1OE 5452 IC50 = 6890 nM T50594 D00IFR 58423153 Ki = 0.017 nM T50594 D02NNV 3038525 IC50 > 5000 nM T50594 D03HUX 49792852 IC50 > 10000 nM T50594 D03ISJ 135564632 IC50 = 42 nM T50594 D07EHV 44814409 Ki = 0.006 nM T50594 D08UUL 46700756 IC50 > 10000 nM T50594 D09JEJ 24748573 IC50 = 46 nM T50594 D0E3TC 44259 IC50 = 2.67 nM T50594 D0G5CS 68071 IC50 = 107000 nM T50594 D0O0LS 25141092 IC50 > 10000 nM T50594 D0O6WV 24794418 IC50 > 2000 nM T50594 D0W3LI 153999 IC50 = 200 nM T50594 D03BNU 59604787 IC50 > 3500 nM T50594 D00OWF 5280953 IC50 > 10000 nM T50594 D04VSB 68356857 IC50 = 5 nM T50594 D06OKX 68356855 IC50 = 4 nM T50594 D08JUU 68327881 IC50 = 15 nM T50594 D0J6HN 46179018 Ki = 0.001 nM T50594 D0M0TH 44480198 IC50 = 660 nM T50594 D0NE0N 44479711 IC50 = 780 nM T50594 D0NS6I 10037501 IC50 > 10000 nM T50594 D0OS2I 59226518 Ki = 0.001 nM T50594 D0P9UF 51002052 Ki < 1 nM T50594 D0Q3VZ 135398522 IC50 = 880 nM T50594 D09SFV 3973 IC50 = 4000 nM T50594 D0T3ME 156422 IC50 > 30000 nM T50594 D0U7OU 3220 IC50 = 2500 nM T50594 C45RGA 10331 IC50 = 119000 nM T50594 C9B1FN 26905 IC50 = 28000 nM T50594 C3EOV0 51082 IC50 = 50.9 nM T50594 CEW91J 72742 IC50 = 21400 nM T50594 CXF8W3 87756 IC50 = 37000 nM T50594 CQB5T6 95731 IC50 = 57100 nM T50594 CV97AF 99135 IC50 = 6730 nM T50594 CA7QS6 99712 IC50 = 8160 nM T50594 CMW74I 294520 IC50 = 6000 nM T50594 CVXN37 313371 IC50 = 7400 nM T50594 CQ32PZ 331313 IC50 = 19200 nM T50594 C3TZJ7 399090 IC50 = 920 nM T50594 C63VHK 456402 IC50 = 2100 nM T50594 CXN6D3 469823 IC50 > 10000 nM T50594 C43QUM 477727 IC50 = 5000 nM T50594 CN6AY0 491467 IC50 = 200 nM T50594 CTFX23 705543 Ki = 3400 nM T50594 CV8C2R 735247 IC50 = 8500 nM T50594 C2O3PU 788302 Ki = 4500 nM T50594 CCPR76 791050 IC50 = 4410 nM T50594 C0KN1S 823103 IC50 = 3000 nM T50594 CP1VI0 848933 IC50 > 20000 nM T50594 C5XGB1 849788 IC50 = 5000 nM T50594 CIW3E8 939111 IC50 = 332 nM T50594 C97VXG 958611 IC50 = 28000 nM T50594 CG5XY6 1201120 IC50 = 45000 nM T50594 C0VOM1 1201137 IC50 = 320 nM T50594 C5PDS4 1206018 IC50 = 600 nM T50594 CQ7PL4 1235170 IC50 = 50 nM T50594 C2REL7 1239884 IC50 = 13 nM T50594 CWU65G 1241133 IC50 = 458 nM T50594 C2JSX4 1241442 IC50 = 890 nM T50594 CFX90H 1243769 IC50 = 650 nM T50594 C97BMP 1307080 IC50 = 12000 nM T50594 C8I0WK 1361334 IC50 = 17 nM T50594 CM3CE2 1379638 IC50 = 40 nM T50594 CIB51E 1379720 IC50 = 130 nM T50594 CR25HA 1379728 IC50 = 10000 nM T50594 CEW8K1 1379922 IC50 = 160 nM T50594 COTN75 1382447 IC50 = 40 nM T50594 C6GN3Z 1526876 IC50 = 62 nM T50594 CWJS81 1539584 IC50 = 950 nM T50594 CB8K9W 1641790 IC50 = 28000 nM T50594 C03SAD 1641793 IC50 = 6000 nM T50594 CK54MC 1750281 IC50 = 386 nM T50594 C7JNA3 1939911 IC50 = 410 nM T50594 CQ7O6N 1963136 IC50 = 388 nM T50594 CH4TI3 2243909 IC50 = 160 nM T50594 C4L6GC 2727417 Ki = 320 nM T50594 C3TJ1I 2765355 Ki = 91 nM T50594 CL2DR0 2816326 IC50 = 3160 nM T50594 CA6M0K 2816444 IC50 = 4790 nM T50594 C8J6MX 2816445 IC50 > 20000 nM T50594 CVGW02 2816447 IC50 = 20000 nM T50594 CHZ0M5 2816450 IC50 = 1230 nM T50594 CGB3K0 2816451 IC50 = 20000 nM T50594 CSWI94 2831986 IC50 = 10000 nM T50594 C9GX8Y 3008939 IC50 = 1000 nM T50594 C8V5MP 3008941 IC50 = 2800 nM T50594 C6HU3T 3008942 IC50 = 600 nM T50594 CLD94C 3008943 IC50 = 3300 nM T50594 C3AD1T 3008944 IC50 = 5100 nM T50594 C7MBD8 3008946 IC50 = 1000 nM T50594 CD47SO 3008947 IC50 = 2000 nM T50594 COQ8W4 3008948 IC50 = 500 nM T50594 CGK6Q2 3157072 IC50 = 63000 nM T50594 CNC5M8 3358971 IC50 = 5800 nM T50594 C02FHS 3497823 IC50 > 20000 nM T50594 CXSP30 3646268 IC50 = 23800 nM T50594 CZ69AG 4119632 IC50 = 3500 nM T50594 CCUW85 4205046 IC50 = 11600 nM T50594 CSF82V 4205283 IC50 = 3600 nM T50594 CRD72J 5003498 Ki = 550 nM T50594 C5XM7Z 5275788 IC50 = 3100 nM T50594 CP29OA 5281628 IC50 = 2710 nM T50594 C8IAR2 5281657 IC50 = 300 nM T50594 CY9C4T 5281680 IC50 = 340 nM T50594 CGF5Q9 5281701 IC50 = 650 nM T50594 CI68PW 5283685 IC50 > 100000 nM T50594 CXK0S6 5283727 IC50 > 100000 nM T50594 C3BW1R 5327669 IC50 = 2000 nM T50594 CNT82G 5327726 IC50 = 150 nM T50594 CFW43H 5340112 IC50 > 10000 nM T50594 C02SGM 5459373 IC50 = 61 nM T50594 CZ0NU2 5481591 IC50 = 55 nM T50594 CDK3J0 5703619 IC50 = 54 nM T50594 C4YEC5 5757257 IC50 = 113 nM T50594 C9DL5A 5878179 IC50 = 170 nM T50594 CH1R8P 5985287 IC50 = 60 nM T50594 C1GZ5L 6006914 IC50 = 330 nM T50594 CAH19P 6026872 IC50 = 600 nM T50594 C4J5VQ 6076476 IC50 = 150 nM T50594 C54UXA 6226569 IC50 = 126 nM T50594 CF06NG 6419809 IC50 = 57 nM T50594 CI0FY2 6475553 IC50 = 3200 nM T50594 C1J4FN 6475556 IC50 = 3400 nM T50594 C50MYS 6475557 IC50 = 4000 nM T50594 CR9Z5I 6475559 IC50 = 400 nM T50594 CLN2G8 6475560 IC50 = 500 nM T50594 C8XYJ1 6479612 IC50 = 3000 nM T50594 C4N3UF 6604030 IC50 = 7030 nM T50594 C3N6ML 6619879 IC50 = 65 nM T50594 CB0V3N 7342915 IC50 = 6700 nM T50594 C4G9WR 9547398 IC50 > 100000 nM T50594 C76CUP 9547698 IC50 > 100000 nM T50594 CY2ZJ8 9840025 Ki = 18 nM T50594 C7GP2B 9965755 IC50 = 67 nM T50594 CW94SP 10016571 Ki = 410 nM T50594 CR8DA1 10024683 IC50 > 100000 nM T50594 CLA93G 10047202 IC50 > 100000 nM T50594 C3LCH5 10047545 IC50 > 100000 nM T50594 C3K7CB 10236138 IC50 = 5300 nM T50594 C7SFI1 10296883 IC50 = 50.12 nM T50594 C8ILG2 10332398 Ki = 1800 nM T50594 CE01GL 10333282 Ki = 210 nM T50594 C6G5TO 10333921 Ki > 3300 nM T50594 C3MC1X 10359460 Ki = 54 nM T50594 CTOQ47 10361208 Ki = 11 nM T50594 CN62MP 10378377 Ki = 430 nM T50594 CRV81H 10401467 Ki = 980 nM T50594 CGJ53E 10423197 Ki > 3300 nM T50594 C4CP7K 10423452 IC50 = 300 nM T50594 C5K2XY 10448624 Ki > 3300 nM T50594 C83QWV 10714343 IC50 = 20300 nM T50594 CMQ86D 10945211 IC50 = 67 nM T50594 CL68JZ 11003572 IC50 = 8700 nM T50594 CTU6W8 11194777 IC50 > 10000 nM T50594 C8G5WP 11210533 IC50 = 4440 nM T50594 CBOP58 11293798 Ki = 1100 nM T50594 C26BZX 11362471 Ki = 280 nM T50594 CWXB93 11397177 Ki > 10000 nM T50594 CTG83F 11539329 Ki > 9200 nM T50594 CACS26 11561968 Ki > 2000 nM T50594 CMIL86 11590363 Ki > 9200 nM T50594 C9T6SC 11640926 Ki > 9200 nM T50594 CP04JC 11666231 IC50 = 103 nM T50594 CU0E8O 11690457 Ki > 2000 nM T50594 CQW78J 11759459 IC50 = 3000 nM T50594 CUE6L3 11782377 IC50 = 4500 nM T50594 C5IR2A 12444300 IC50 = 7390 nM T50594 CDFI41 13365773 IC50 = 7800 nM T50594 CCG79O 13814386 IC50 = 20 nM T50594 CFPW41 16007116 Ki > 9200 nM T50594 COPQ34 16043794 Ki = 15 nM T50594 CW2XK6 16050925 IC50 = 340 nM T50594 CGC34R 16118737 IC50 > 30000 nM T50594 C5VPH9 16129448 IC50 > 10000 nM T50594 CH1G2J 16348526 IC50 = 6.7 nM T50594 CY1E2N 16723801 IC50 > 100000 nM T50594 CH1ZG4 17129569 IC50 = 55 nM T50594 C0SQ8M 17404949 IC50 = 11 nM T50594 C5LIA8 18965707 IC50 > 10000 nM T50594 CBG4X2 20784957 Ki = 3300 nM T50594 C76BQI 20877991 IC50 = 14 nM T50594 CZMD21 20877999 IC50 = 96 nM T50594 CDK8B0 21443955 IC50 = 371 nM T50594 CN2J6M 21964150 IC50 = 6100 nM T50594 CV1LT2 23770859 IC50 = 50 nM T50594 CG0NS1 24737654 IC50 = 13 nM T50594 C7YG1N 24759534 IC50 = 590 nM T50594 CQNP54 24764449 IC50 = 25000 nM T50594 C4Z9CN 24769780 IC50 = 7800 nM T50594 CP1WR0 24795070 IC50 = 7 nM T50594 CLCU03 24811585 IC50 = 33 nM T50594 C0K7NB 24811691 IC50 = 370 nM T50594 CY8X0J 24811794 IC50 = 57 nM T50594 C73WEX 24812008 IC50 = 50 nM T50594 C4D2QE 24894053 Ki = 0.002 nM T50594 CY8L7E 24896769 IC50 > 10000 nM T50594 C1XI6G 25025645 IC50 = 18 nM T50594 CX1HL8 25032704 Ki = 2.5 nM T50594 CB21XV 25164469 Ki > 8570 nM T50594 CNF0A8 25164674 Ki = 3685 nM T50594 CUX83H 25164675 Ki > 8570 nM T50594 C1H7BF 25164677 Ki > 8570 nM T50594 CN50EI 25164678 Ki > 8750 nM T50594 C3XI7P 25164880 Ki > 8750 nM T50594 CX80QK 25164883 Ki = 339 nM T50594 C6SD2A 25165081 Ki > 8570 nM T50594 C67TVH 25165085 Ki > 8570 nM T50594 C8J4KL 25165278 Ki = 5155 nM T50594 CRJ6M7 25165279 Ki > 8750 nM T50594 C7RBX0 25165280 Ki > 8750 nM T50594 CPEY29 25165481 Ki > 8750 nM T50594 C70DRX 25165482 Ki > 8750 nM T50594 CE8D1W 25165860 Ki = 2219 nM T50594 C6VZU2 25165861 Ki = 923 nM T50594 C9VA1N 25166056 Ki = 10153 nM T50594 C1JS9O 25166057 Ki = 12000 nM T50594 CM41PX 25166058 Ki = 165230 nM T50594 CT94MS 25166059 Ki = 4153 nM T50594 CCN25J 25166251 Ki = 37846 nM T50594 CX8HY9 25166657 Ki = 20307 nM T50594 C1CNX7 25166659 Ki = 36000 nM T50594 C81WIV 25166867 Ki = 41538 nM T50594 C9MR2O 25166869 Ki = 1292 nM T50594 CAG1H6 25166870 Ki = 2307 nM T50594 CFE4O7 25166871 Ki = 1846 nM T50594 CGUC69 25167072 Ki = 307 nM T50594 CF4G1L 25167074 Ki = 242 nM T50594 C35ZXL 25167075 Ki = 2656 nM T50594 C1CRJ7 25167076 Ki = 4156 nM T50594 C1IFX5 25167077 Ki = 1952 nM T50594 C2D3FP 25167078 Ki > 8750 nM T50594 CP2W8I 25167079 Ki = 2899 nM T50594 CJO5A4 25167275 Ki > 8750 nM T50594 C5KX0G 25167277 Ki = 114 nM T50594 CQ5FJ8 25167278 Ki > 8750 nM T50594 C37YSX 25167280 Ki = 1664 nM T50594 C4ZQ9E 25169520 IC50 = 8000 nM T50594 CS2P3O 25185171 IC50 = 73 nM T50594 CLG79A 25185172 IC50 = 69000 nM T50594 C90BFN 25185173 IC50 = 73000 nM T50594 CMI7T4 25185174 IC50 = 58000 nM T50594 CLH4S6 25185175 IC50 = 78000 nM T50594 C3QF7Z 25185441 IC50 = 28000 nM T50594 C0R4PY 25185442 IC50 = 45000 nM T50594 C19MTD 25185443 IC50 = 38000 nM T50594 CO6L0V 25185444 IC50 = 78000 nM T50594 CDN2V4 25189319 IC50 = 460 nM T50594 C2DSU0 25189321 IC50 = 280 nM T50594 C46UKS 25189322 IC50 = 300 nM T50594 CQ53XH 25190443 Ki = 11 nM T50594 C3ZH2Q 25190444 IC50 = 340 nM T50594 C64HVI 25190445 IC50 = 370 nM T50594 CF4BU7 25190446 IC50 = 430 nM T50594 CCKG72 25190447 IC50 = 1030 nM T50594 CL5RN6 25190448 IC50 = 1140 nM T50594 C08EZS 25190451 IC50 > 20000 nM T50594 C7IR2T 25190452 IC50 > 20000 nM T50594 CIY3A2 25190453 Ki = 21.8 nM T50594 CN0YI4 25190454 Ki = 12.3 nM T50594 C0YXD8 25190455 Ki = 15 nM T50594 CC10AL 25190456 Ki = 36.5 nM T50594 CHP23Y 25190458 Ki = 1271 nM T50594 CIWV65 25190459 Ki = 271 nM T50594 C1KY2L 25190460 Ki = 4894 nM T50594 C19AOI 25190461 Ki = 1162 nM T50594 C8V0PL 25190462 Ki = 2698 nM T50594 CL85GI 39005031 Ki = 90 nM T50594 CIKM57 44180156 IC50 = 43 nM T50594 CB0O2A 44186880 Ki > 8570 nM T50594 C9K7OP 44186882 Ki = 8359 nM T50594 CX0ZU8 44186885 Ki > 8570 nM T50594 CUQE83 44187007 IC50 = 2 nM T50594 CNGV37 44189584 Ki > 8570 nM T50594 C9V3XY 44199470 Ki = 0.01 nM T50594 CU13JS 44217530 Ki < 1 nM T50594 CW96TZ 44217683 Ki < 1 nM T50594 C8KNA3 44219632 Ki = 21 nM T50594 C0VIX4 44219633 Ki < 5 nM T50594 CBW35D 44222957 IC50 = 27 nM T50594 C0LDV8 44222965 IC50 = 5 nM T50594 C3ZJ6S 44222969 IC50 = 4 nM T50594 CX4SQ0 44222970 IC50 = 2 nM T50594 CAG56N 44222977 IC50 = 7 nM T50594 CPJ3G8 44241505 IC50 = 120 nM T50594 CS89EN 44479467 IC50 = 570 nM T50594 C03IGD 44540030 IC50 = 1995.26 nM T50594 C5LWU1 44540126 IC50 = 2511.89 nM T50594 C2T9GC 44540407 IC50 = 2511.89 nM T50594 CQ4PE7 44540492 IC50 = 15848.93 nM T50594 CL3M2Q 44545852 Ki = 5 nM T50594 CAR15E 44573514 IC50 = 120 nM T50594 C5A3IV 44573834 Ki = 44 nM T50594 CBG03H 44573835 Ki = 94 nM T50594 CG42VU 44573866 Ki = 160 nM T50594 C23QJX 44573945 Ki = 49 nM T50594 C04QEC 44573946 Ki = 100 nM T50594 C2NCR5 44574367 Ki = 50 nM T50594 C01GEN 44581101 IC50 = 75000 nM T50594 CU7QD2 44582386 IC50 = 2100 nM T50594 COY57J 44592504 IC50 = 794 nM T50594 CID7A6 44593656 IC50 = 4000 nM T50594 CEQN62 44609163 IC50 < 3 nM T50594 C7G4FT 44609164 IC50 < 3 nM T50594 CH9FO5 44609165 IC50 < 3 nM T50594 CLPY85 44609168 IC50 < 3 nM T50594 CU0QT2 44609322 IC50 < 3 nM T50594 CQ06VN 44609327 IC50 < 3 nM T50594 CE9GN6 44609485 IC50 = 9 nM T50594 C4QC7B 44609634 IC50 = 36 nM T50594 C37RDC 45110412 IC50 = 73 nM T50594 CV7S5L 45110413 IC50 = 41 nM T50594 CU3RF1 45139989 IC50 > 10000 nM T50594 CQGZ06 45139991 IC50 > 10000 nM T50594 CDS4J9 46178380 Ki < 1 nM T50594 CP0WY1 46178460 Ki = 5 nM T50594 C8Y2OV 46178825 IC50 = 11 nM T50594 C4S8MP 46179491 Ki < 1 nM T50594 CY3HW5 46224684 IC50 = 1400 nM T50594 CDQ1K4 46224842 IC50 = 50000 nM T50594 C7ON5A 46233287 IC50 > 10000 nM T50594 CLS29B 46872626 IC50 > 10000 nM T50594 C2O8RZ 46886323 IC50 > 1000 nM T50594 CA86TF 46887815 IC50 > 10000 nM T50594 C5UHD4 46887816 IC50 > 10000 nM T50594 C89JAV 46887868 IC50 > 10000 nM T50594 CZ32AN 46887899 IC50 > 10000 nM T50594 CQI2Y6 46887900 IC50 = 5000 nM T50594 CCN08S 46934144 IC50 > 100000 nM T50594 C09RXA 46937301 IC50 = 6.8 nM T50594 CPW9Z5 46937316 IC50 = 31 nM T50594 C2HZ3M 49779260 IC50 = 12 nM T50594 CAZ1V8 49805556 IC50 = 38 nM T50594 CF91RS 49843531 IC50 > 10000 nM T50594 CVQ6P3 50915164 IC50 = 3 nM T50594 C68POW 50941395 IC50 = 342 nM T50594 CF3YB2 50941397 IC50 = 577 nM T50594 CX93HP 50942535 IC50 > 2500 nM T50594 C71RUL 50942628 IC50 > 2500 nM T50594 CZ8B9T 50942630 IC50 = 798 nM T50594 CUG03K 51033838 IC50 = 1 nM T50594 C5NT2O 51036049 IC50 = 7 nM T50594 CK0MX5 51036250 IC50 = 5 nM T50594 C4RH7Z 51036450 IC50 = 2 nM T50594 C1RN8T 51036645 IC50 = 2 nM T50594 CO7MY6 51036646 IC50 = 9 nM T50594 CEG98T 51036856 IC50 = 15 nM T50594 C7B1JO 51037081 IC50 = 16 nM T50594 CDTC84 51037916 IC50 = 4 nM T50594 CDU4Q5 51346827 Ki > 8570 nM T50594 C4PI9Q 51351831 IC50 = 120 nM T50594 CG5IK8 52936268 IC50 > 31600 nM T50594 COW1J0 52936347 IC50 = 40000 nM T50594 CEQN27 52936621 Ki > 1000 nM T50594 C60WAG 52940742 IC50 = 66 nM T50594 CA3FI5 52943221 IC50 = 18 nM T50594 CR7A0Z 52945651 IC50 = 30 nM T50594 C3DTV5 53233133 IC50 = 20 nM T50594 C2CT5J 53236670 IC50 > 100000 nM T50594 C3M6LV 53236671 IC50 > 31600 nM T50594 CZ5L6F 53239373 IC50 = 37100 nM T50594 C2WFI8 53239374 IC50 > 100000 nM T50594 C0ZHF8 53239375 IC50 > 100000 nM T50594 CD1EQ3 53239587 IC50 = 32540 nM T50594 C82IWE 53250611 IC50 = 400 nM T50594 C1XP7K 53308973 IC50 > 10000 nM T50594 CBPV19 53308974 IC50 = 7000 nM T50594 C58TBY 53308976 IC50 = 4000 nM T50594 C2CH7R 53309118 IC50 = 4100 nM T50594 CDV5X6 53309119 IC50 > 10000 nM T50594 C2QW5D 53309120 IC50 = 2200 nM T50594 CZS8K4 53319042 Ki > 8570 nM T50594 CUD21V 53320263 Ki > 8570 nM T50594 CESA85 53323614 Ki > 8570 nM T50594 CNPM14 53341082 IC50 > 3000 nM T50594 CM98WS 53372413 IC50 > 10000 nM T50594 CM0QI9 53372414 IC50 = 69 nM T50594 CH70WB 53372416 IC50 = 316 nM T50594 C3HU1Q 53372540 IC50 = 155 nM T50594 CNI7P9 53372541 EC50 = 45 nM T50594 C0IYG7 53372543 IC50 = 17 nM T50594 C8F0JA 53372544 IC50 = 10 nM T50594 CA6H2P 53372668 IC50 = 6 nM T50594 CY1I9B 53372669 IC50 = 11 nM T50594 COP26H 53372670 IC50 = 4 nM T50594 CFM7W8 53372672 IC50 = 1.5 nM T50594 C9GYZ3 53372790 IC50 = 1 nM T50594 C8BP9G 53372791 IC50 = 266 nM T50594 CXM10V 53372792 IC50 = 238 nM T50594 C8NA4L 53384644 IC50 > 30000 nM T50594 C49DRM 53482602 Ki = 0.02 nM T50594 CS4Y9F 53482665 Ki = 0.6 nM T50594 CR9P7C 53482785 Ki = 0.2 nM T50594 C5IWB4 53482960 Ki = 0.09 nM T50594 CBS73R 53484203 Ki = 6500 nM T50594 C43MFC 54576041 IC50 = 2 nM T50594 C2AJ9L 54576042 IC50 = 2 nM T50594 CQFH98 54580157 IC50 = 7400 nM T50594 CR1UO2 54580158 IC50 = 450 nM T50594 CA43ED 54581151 IC50 = 6000 nM T50594 C3H9FS 54581152 IC50 = 460 nM T50594 C56PNV 54581153 IC50 = 53 nM T50594 CG4FR6 54581154 IC50 = 60 nM T50594 C75IDW 54581155 IC50 = 4500 nM T50594 C9IL8D 54581156 IC50 = 150 nM T50594 C3N8XT 54581186 IC50 = 2300 nM T50594 CVNC57 54582208 IC50 = 2700 nM T50594 C0TZ7R 54583142 IC50 = 210 nM T50594 C73GAJ 54583143 IC50 = 51 nM T50594 C1NLW0 54585070 IC50 = 71 nM T50594 CJO3M1 54585071 IC50 = 55 nM T50594 CN73GO 54585072 IC50 = 220 nM T50594 CH6CE1 54586044 IC50 = 380 nM T50594 CF7B2S 54586045 IC50 = 1900 nM T50594 CYD87G 54586046 IC50 = 4900 nM T50594 CI9U5M 54586075 IC50 = 980 nM T50594 CH03RW 54587027 IC50 = 5400 nM T50594 CL38AX 54587028 IC50 = 40 nM T50594 C6Q7BN 54691404 IC50 = 17000 nM T50594 CWQ31J 54752779 IC50 < 2 nM T50594 CZ4CR6 54752780 IC50 < 2 nM T50594 C96CIG 54752781 IC50 < 2 nM T50594 C2FK8I 54752782 IC50 < 2 nM T50594 C9ZFS1 54764923 IC50 > 100000 nM T50594 CM8JX1 56604907 IC50 = 25000 nM T50594 CAR67O 56665753 Ki = 11500 nM T50594 CC7T2A 56674921 IC50 = 170 nM T50594 CLHO15 56676037 Ki = 6600 nM T50594 CFB2R8 56676630 IC50 = 2600 nM T50594 CN8YK1 56935642 IC50 = 28 nM T50594 C1JLW8 57332840 IC50 = 2610 nM T50594 CD01JZ 57332841 IC50 = 8300 nM T50594 CCFK37 57332844 IC50 = 2830 nM T50594 CK1SR7 57332969 IC50 = 4400 nM T50594 C5TRE2 57332970 IC50 = 8570 nM T50594 C46TJK 57332974 IC50 = 31200 nM T50594 C09ZJY 57333095 IC50 = 11340 nM T50594 CWQP86 57342345 IC50 = 0.47 nM T50594 CFKA67 57390288 IC50 = 192 nM T50594 CYF74P 57390289 IC50 = 2100 nM T50594 C4Y3WA 57390290 IC50 < 2 nM T50594 CU3WM8 57390291 IC50 = 17 nM T50594 CGT82N 57390292 IC50 = 23 nM T50594 CO92HZ 57390346 IC50 = 8 nM T50594 CC3X4H 57390347 IC50 = 41 nM T50594 C9J5YZ 57391268 IC50 = 217 nM T50594 CV6DG1 57391610 IC50 = 400 nM T50594 C1Y2OG 57391625 IC50 = 77 nM T50594 CIHG14 57391626 IC50 = 126 nM T50594 CUB01N 57391627 IC50 = 133 nM T50594 CS0Y1G 57392065 IC50 = 2500 nM T50594 C13ARH 57392066 IC50 = 11000 nM T50594 CAD9Q1 57392067 IC50 = 194 nM T50594 CD7R3C 57392125 IC50 = 7 nM T50594 CG5LM0 57392126 IC50 = 9 nM T50594 C53YDP 57392127 IC50 = 8 nM T50594 CZT5Q4 57392128 IC50 = 24 nM T50594 C1LDX8 57393366 IC50 = 3260 nM T50594 CD3Z8R 57393367 IC50 = 68 nM T50594 CUWX39 57393368 IC50 = 2420 nM T50594 CGHN79 57393369 IC50 = 14 nM T50594 C1SGW3 57393817 IC50 = 15000 nM T50594 C34RIH 57393818 IC50 = 250 nM T50594 C6I5MD 57393819 IC50 = 107 nM T50594 C6ZNF8 57393820 IC50 = 228 nM T50594 CT2IK5 57393821 IC50 = 52 nM T50594 C24ITU 57393822 IC50 = 28 nM T50594 C1K4BX 57393824 IC50 = 45 nM T50594 CYK23D 57393887 IC50 = 55 nM T50594 CHG95S 57393892 IC50 = 10 nM T50594 CA28OK 57393893 IC50 = 16 nM T50594 C6PN4T 57393894 IC50 = 25 nM T50594 C2WR6L 57395087 IC50 = 2600 nM T50594 CA7PC1 57395088 IC50 = 165 nM T50594 C29ZPK 57395544 IC50 = 4 nM T50594 CWV27Q 57395545 IC50 = 110 nM T50594 CGJ67T 57395546 IC50 = 39 nM T50594 C04UWN 57395547 IC50 = 41 nM T50594 CQEL83 57395548 IC50 = 74 nM T50594 C82EYJ 57395549 IC50 = 26 nM T50594 CXN51F 57395611 IC50 = 2220 nM T50594 CS4Q7E 57395612 IC50 > 2500 nM T50594 C42ESL 57395623 IC50 = 16 nM T50594 CL58MG 57395624 IC50 = 21 nM T50594 CSZ37K 57396179 IC50 = 2600 nM T50594 CE2YT1 57396291 IC50 = 13 nM T50594 C06LDJ 57396331 IC50 = 105 nM T50594 CW4KG3 57396858 IC50 = 9 nM T50594 CA2G6Z 57396964 IC50 = 282 nM T50594 CIBU80 57397370 IC50 = 4900 nM T50594 CC6Q2N 57397371 IC50 < 2 nM T50594 CNC93S 57397372 IC50 = 7 nM T50594 C0F3LV 57397435 IC50 = 8 nM T50594 C70URD 57397436 IC50 = 13 nM T50594 C1UZP2 57397437 IC50 = 10 nM T50594 C1L4HY 57398127 IC50 = 8 nM T50594 C87MDQ 57398621 IC50 = 433 nM T50594 C5NOH0 57398622 IC50 = 35 nM T50594 C9GP1C 57398623 IC50 = 844 nM T50594 CODG52 57398624 EC50 = 380 nM T50594 CDBZ51 57398625 IC50 = 317 nM T50594 C0PNU8 57399041 IC50 = 25 nM T50594 C1NLS0 57399688 IC50 = 327 nM T50594 C0YAL9 57399780 IC50 = 315 nM T50594 C7RF5J 57399974 IC50 = 25 nM T50594 CQ5YP2 57399976 IC50 = 79 nM T50594 CFRP21 57400282 IC50 = 162 nM T50594 CHP7S8 57400283 IC50 = 226 nM T50594 C4CW2G 57400284 IC50 = 38 nM T50594 C1E2UR 57400285 IC50 = 87 nM T50594 CL1W3P 57400286 IC50 = 336 nM T50594 C91XMS 57400287 IC50 = 405 nM T50594 CC73VO 57400785 IC50 = 2800 nM T50594 CM7NS6 57400786 IC50 < 2 nM T50594 CX5MH0 57400787 IC50 < 2 nM T50594 CD47VK 57400788 IC50 = 114 nM T50594 CR29GW 57400789 IC50 = 13 nM T50594 C3G5BY 57400790 IC50 = 21 nM T50594 CAD5G6 57400791 IC50 = 26 nM T50594 C6QIJ2 57400845 IC50 > 2500 nM T50594 C9NJ0A 57400853 IC50 = 6 nM T50594 CM24WI 57400854 IC50 = 2 nM T50594 CJ4YR1 57400855 IC50 = 7 nM T50594 CP80OE 57402076 IC50 = 108 nM T50594 C36ZSI 57402544 IC50 = 1700 nM T50594 C6F9HJ 57402545 IC50 = 170 nM T50594 CVBS23 57402546 IC50 = 530 nM T50594 CG35HA 57402547 IC50 < 2 nM T50594 CW7I5C 57402548 IC50 = 18 nM T50594 C9GXO5 57402606 IC50 = 100 nM T50594 CT5F2M 57403491 IC50 = 127 nM T50594 CIV6R9 57403842 IC50 = 852 nM T50594 CIQT05 57403843 IC50 = 320 nM T50594 C8F6AY 57403844 IC50 = 436 nM T50594 CA71NH 57403845 IC50 = 5 nM T50594 CK6H4W 57403939 IC50 = 3910 nM T50594 CZSM95 57412684 IC50 > 10000 nM T50594 C6JET5 58182164 Ki = 0.04 nM T50594 CPU40N 58189477 IC50 = 8 nM T50594 C2B4KD 58189484 IC50 = 91 nM T50594 CGML85 58189493 IC50 = 11 nM T50594 C4PI2X 58189496 IC50 = 15 nM T50594 CL85RA 58189505 IC50 = 16 nM T50594 CD96SU 58189506 IC50 = 17 nM T50594 C3J0BF 58189523 IC50 = 64 nM T50594 C3ZAY9 58189525 IC50 = 9 nM T50594 C1QM9E 58189526 IC50 = 4 nM T50594 CL5J0G 58189527 IC50 = 14 nM T50594 C6P8JQ 58189528 IC50 = 6 nM T50594 C3X1OD 58189540 IC50 = 69 nM T50594 CCJW98 58189542 IC50 = 10 nM T50594 C63GUR 58189549 IC50 = 4 nM T50594 CP12HS 58189553 IC50 = 27 nM T50594 CI8QG4 58189555 IC50 = 9 nM T50594 CP3YX7 58189559 IC50 = 14 nM T50594 CE96XT 58189563 IC50 = 5 nM T50594 CL3AQ9 58189570 IC50 = 6 nM T50594 CLB8X2 58189576 IC50 = 3 nM T50594 C37EVM 58189578 IC50 = 5 nM T50594 CO87KC 58189587 IC50 = 7 nM T50594 CL5R9Q 58189614 IC50 = 4 nM T50594 CJ9RY1 58189624 IC50 = 16 nM T50594 C8GU4K 58189625 IC50 = 17 nM T50594 CO06IF 58189629 IC50 = 4 nM T50594 C78RDU 58189641 IC50 = 35 nM T50594 C6C4FH 58313037 Ki = 7.7 nM T50594 CXT6Q2 58423155 IC50 = 28 nM T50594 C73BEA 58423187 IC50 = 1500 nM T50594 C3KL4R 58423251 IC50 = 18 nM T50594 CF0L6E 58423275 IC50 < 6 nM T50594 CY2I5D 58423319 IC50 = 12 nM T50594 CBY0I7 58423384 IC50 = 61 nM T50594 CRG4K0 58464982 Ki = 0.08 nM T50594 CS4GX1 58826480 IC50 = 833 nM T50594 CLE79F 59190121 IC50 = 25 nM T50594 CW7F1B 59190170 IC50 = 45 nM T50594 CS4Y8U 59190179 IC50 = 43 nM T50594 CC3HF5 59190198 IC50 = 21 nM T50594 CEI9F1 59190242 IC50 = 506 nM T50594 C4T8QV 59190250 IC50 = 74.4 nM T50594 C7E3JK 59190306 IC50 = 3 nM T50594 C6H8IU 59226389 Ki < 1 nM T50594 C0K9MU 59380314 IC50 = 52000 nM T50594 CCU1I6 59455685 Ki < 1 nM T50594 C4KV1J 59587678 IC50 = 8 nM T50594 CGV9W1 59587708 IC50 = 14 nM T50594 CXJ63M 59603829 IC50 = 9900 nM T50594 CQEU96 59603842 IC50 = 2800 nM T50594 C16YEO 59662448 IC50 = 82 nM T50594 CPR84X 59662532 IC50 = 18 nM T50594 C1MR8Q 60097495 IC50 > 1000 nM T50594 CV49AH 60155621 IC50 = 102 nM T50594 CPN9Z7 60155622 IC50 = 17 nM T50594 CB6PX9 60155697 IC50 = 6 nM T50594 CQ0J1X 60155698 IC50 = 12 nM T50594 CH4NS1 60155699 IC50 = 43 nM T50594 C9V2EM 60155700 IC50 = 92 nM T50594 C5AQ6G 60155701 IC50 = 53 nM T50594 C1C4BG 60155702 IC50 = 447 nM T50594 CK9B3E 60155783 IC50 = 20 nM T50594 C8SLY4 60168156 IC50 = 46 nM T50594 C57MNF 60168157 IC50 = 470 nM T50594 CFB45M 60168158 IC50 = 75 nM T50594 CI4NU3 60459498 IC50 = 21 nM T50594 C4BRH3 62046501 Ki = 1800 nM T50594 C90ZFG 66597948 IC50 = 204 nM T50594 CHO3M7 66597981 IC50 = 27 nM T50594 CYO8V7 66597989 IC50 = 148 nM T50594 C7W2XF 66597997 IC50 = 23 nM T50594 C16DNF 66598062 IC50 = 24 nM T50594 CMA92Y 66598080 Ki = 5 nM T50594 C4RCD5 66598081 IC50 = 5 nM T50594 C38XNO 66598093 IC50 = 132 nM T50594 C52HRW 66598095 IC50 = 25 nM T50594 C82RIS 66598100 IC50 = 164 nM T50594 CRDF75 66598125 IC50 = 111 nM T50594 CF9T4M 66598126 IC50 = 237 nM T50594 C1ET4P 66598128 IC50 = 45 nM T50594 C5D3TJ 66598153 IC50 = 17 nM T50594 CJFZ71 66598162 IC50 = 197 nM T50594 CG7X8T 66598186 IC50 = 54 nM T50594 CF5R9E 66598190 IC50 = 378 nM T50594 CBS45L 66615214 IC50 = 68 nM T50594 C8LT0N 66615220 IC50 = 66 nM T50594 CJ31XD 66615233 IC50 = 378 nM T50594 CX8T5L 66772114 IC50 = 57 nM T50594 C37NKO 67129970 IC50 = 1360 nM T50594 CK80LJ 67130050 IC50 > 10000 nM T50594 CNXU89 67162253 IC50 < 500 nM T50594 CV63UL 67240318 IC50 > 10000 nM T50594 C7FCH0 67959600 IC50 = 7 nM T50594 CB65ES 67959736 IC50 = 2 nM T50594 CTK1D8 67959952 IC50 = 15 nM T50594 CE54CI 67960005 IC50 = 127 nM T50594 CY3AZ9 67960061 IC50 = 0.4 nM T50594 CV8O1G 67960139 IC50 = 3 nM T50594 CVFC41 67960161 IC50 = 8 nM T50594 CP2G8D 67960181 IC50 = 1 nM T50594 CR7DN8 68032650 IC50 = 5 nM T50594 CGO14Q 68161034 Ki < 1 nM T50594 C02UIN 68161275 Ki = 18 nM T50594 C4XZ5Q 68161316 Ki = 810 nM T50594 CA0UR4 68161594 Ki = 6 nM T50594 CY0QN9 68161639 Ki = 122 nM T50594 CD41ZA 68161763 Ki = 11 nM T50594 C0US3B 68161865 Ki = 17 nM T50594 C36FUI 68161871 Ki < 1 nM T50594 CYJQ86 68162030 Ki = 28 nM T50594 C6FEN2 68162062 Ki = 2 nM T50594 CJR94B 68162223 Ki = 8 nM T50594 CAD7C0 68162522 Ki = 4 nM T50594 C9GJN4 68162758 Ki = 56 nM T50594 C09NJI 68162802 Ki < 1 nM T50594 C57KXW 68162851 Ki = 4 nM T50594 C97XLW 68163204 Ki < 1 nM T50594 C1E3XF 68184638 Ki < 1 nM T50594 C3SFB2 68184734 Ki = 1 nM T50594 C9XD8R 68187352 Ki < 1 nM T50594 CH2FV7 68187375 Ki = 0.03 nM T50594 CN6A5W 68187418 Ki < 1 nM T50594 CYM62W 68187421 Ki = 16 nM T50594 CYR6N1 68187478 Ki < 1 nM T50594 C7YX8H 68187480 Ki < 1 nM T50594 CKD38R 68187493 Ki = 3 nM T50594 CU3L1D 68187495 Ki < 1 nM T50594 CY6CG5 68187593 Ki < 1 nM T50594 CUB29K 68187641 Ki < 1 nM T50594 C4VUW2 68328157 IC50 = 1020 nM T50594 CA19JZ 68328195 IC50 = 21 nM T50594 CC5F2N 68328262 IC50 = 2740 nM T50594 CDP01I 68328283 IC50 = 17 nM T50594 CA1NW4 68328307 IC50 = 1 nM T50594 C2PK9C 68328329 IC50 = 16 nM T50594 CM5NV2 68328390 IC50 = 48 nM T50594 COQ2P8 68328395 IC50 = 11 nM T50594 CRT84L 68328588 IC50 = 12 nM T50594 CGP7B8 68328695 IC50 = 177 nM T50594 C67HDR 68328735 IC50 = 109 nM T50594 C7O9RP 68356711 IC50 = 8 nM T50594 C7GRD4 68356716 IC50 = 7 nM T50594 CYP10F 68356783 IC50 = 865 nM T50594 CQ6VX1 68356838 IC50 = 24 nM T50594 CUKO28 68356850 IC50 = 142 nM T50594 C4JR8X 68356863 IC50 = 272 nM T50594 C7GRV2 68755406 IC50 > 10000 nM T50594 C5DGR9 69036886 IC50 = 10000 nM T50594 CT8O2I 69042864 Ki = 0.002 nM T50594 CSD25R 69045198 Ki = 3 nM T50594 C5NL7W 69047229 Ki < 1 nM T50594 CXI31L 69047447 Ki = 30 nM T50594 C6QXP3 69090096 Ki < 1 nM T50594 C7B1IP 69090444 Ki < 1 nM T50594 CRBN93 70687077 IC50 = 3000 nM T50594 CS08NG 70692246 Ki = 11 nM T50594 CBJF23 70692372 IC50 = 131 nM T50594 C3O8YB 70694431 IC50 = 67 nM T50594 CVA08R 70696405 IC50 = 91 nM T50594 CAMN71 70696496 IC50 = 21 nM T50594 C3GDX9 70696694 IC50 < 3 nM T50594 CMAT40 70981556 IC50 = 569 nM T50594 C7DO2P 70981589 IC50 = 0.89 nM T50594 C0WC3B 70981821 IC50 = 0.38 nM T50594 C23ARZ 70982089 IC50 = 0.23 nM T50594 C0Y8PA 70982249 IC50 = 56 nM T50594 CNKX61 70982376 IC50 = 1 nM T50594 CH7J2X 70982568 IC50 = 0.024 nM T50594 CM4T3D 70983036 IC50 = 0.26 nM T50594 C97WBL 70983181 IC50 = 0.035 nM T50594 C61DAP 70983443 IC50 = 0.06 nM T50594 C9ASG6 70984064 IC50 = 0.07 nM T50594 CVT09B 71007225 IC50 = 2.9 nM T50594 C1BND0 71007226 IC50 = 0.78 nM T50594 C35VQT 71007233 IC50 = 0.94 nM T50594 C0O7XS 71007248 IC50 = 0.23 nM T50594 CFD27U 71007268 IC50 > 1000 nM T50594 CWK3P9 71007275 IC50 = 3.7 nM T50594 C17CSR 71007292 IC50 = 2 nM T50594 CT23JC 71007294 IC50 = 0.51 nM T50594 C5DA2P 71007297 IC50 = 7.6 nM T50594 C34ANW 71007298 IC50 = 0.062 nM T50594 CG9L5B 71007300 IC50 = 30 nM T50594 CILG13 71007335 IC50 = 1.8 nM T50594 C2K6EB 71007339 IC50 = 1.5 nM T50594 CZ1TG7 71007340 IC50 = 0.39 nM T50594 CR1G6M 71007342 IC50 = 2.2 nM T50594 C0KEC3 71007349 IC50 = 0.83 nM T50594 CBF2N4 71007352 IC50 = 19 nM T50594 C0XZ4A 71007357 IC50 = 10 nM T50594 CO3C5Z 71007358 IC50 = 7.4 nM T50594 C2WF8G 71202406 EC50 = 5360 nM T50594 CCN94X 71227735 IC50 = 94 nM T50594 C4IEN5 71253342 Ki = 0.04 nM T50594 C6VHC3 71253383 Ki = 0.013 nM T50594 C3EF9T 71253391 Ki = 0.021 nM T50594 CQI4F0 71253507 Ki = 13 nM T50594 C8NX5J 71253513 Ki = 0.27 nM T50594 C9I2AE 71253517 Ki = 2 nM T50594 CTR6B1 71253520 Ki = 14 nM T50594 CP4SE3 71253554 Ki = 0.04 nM T50594 CH9RZ3 71253640 Ki = 0.6 nM T50594 CIN75X 71253646 Ki = 10 nM T50594 CI4BD1 71253671 Ki = 0.073 nM T50594 CU1QK9 71253681 Ki = 0.015 nM T50594 CZ9DL0 71253684 Ki = 10 nM T50594 CZA1B4 71253727 Ki = 0.22 nM T50594 CDJ29S 71253734 Ki = 0.036 nM T50594 CX7Z3V 71253771 Ki = 0.06 nM T50594 CPLG04 71253796 Ki = 0.041 nM T50594 C8YOC3 71253802 Ki = 3.3 nM T50594 C6QV8R 71253835 Ki = 0.14 nM T50594 CQL89K 71253906 Ki = 0.035 nM T50594 C6YKF5 71253921 Ki = 7.7 nM T50594 CUBE27 71253945 Ki = 6 nM T50594 CP60UQ 71253958 Ki = 0.3 nM T50594 CWRX87 71254005 Ki = 4 nM T50594 CCNF28 71254040 Ki = 3500 nM T50594 CJTH24 71254053 Ki = 171 nM T50594 CW8H0Y 71254055 Ki = 200 nM T50594 C1W5TL 71254066 Ki = 0.39 nM T50594 COM7L3 71254090 Ki = 0.02 nM T50594 CBST91 71254178 Ki = 0.01 nM T50594 C1HB5Q 71254188 Ki = 0.022 nM T50594 C4GTF2 71254199 Ki = 0.3 nM T50594 CB7Z5W 71254288 Ki = 0.1 nM T50594 CA8G2O 71254348 Ki = 1.82 nM T50594 C2CJI8 71254349 Ki = 31 nM T50594 C2HKV3 71262574 IC50 = 1 nM T50594 C6RA0F 71262581 IC50 = 1 nM T50594 C9QE2L 71262654 IC50 = 5 nM T50594 C2OA1S 71262676 IC50 = 4 nM T50594 CS3E8P 71262754 IC50 = 1 nM T50594 C90JDF 71262764 IC50 = 1 nM T50594 CP0GU5 71262790 IC50 = 28 nM T50594 CZ89GY 71262793 IC50 = 4 nM T50594 C5DXK1 71307955 Ki = 0.003 nM T50594 CKT60L 71455860 Ki = 1600 nM T50594 C8Y3VW 71465328 IC50 = 0.15 nM T50594 C0LI2T 71488479 EC50 = 700 nM T50594 CE41DB 71488550 EC50 = 1380 nM T50594 CJR9V5 71488552 IC50 = 38 nM T50594 CT2L4I 71512722 Ki = 300 nM T50594 CZR1K3 71533687 IC50 = 1 nM T50594 C1SM3T 71539661 Ki = 0.005 nM T50594 CX4JZ9 71547606 IC50 = 530 nM T50594 C2T8KH 71547773 IC50 = 5 nM T50594 CCN01X 71547862 IC50 = 30 nM T50594 CIRD52 71547864 IC50 = 26 nM T50594 CM26ER 71547948 IC50 = 13 nM T50594 CC34DW 71547950 IC50 = 9 nM T50594 CRX81Q 71575642 IC50 > 10000 nM T50594 CZK04P 71580780 IC50 = 230 nM T50594 CW08ZH 71580788 IC50 = 460 nM T50594 C6AN7B 71624486 Ki = 1.1 nM T50594 CJ4S3H 71624487 Ki = 0.052 nM T50594 CL5SN0 71624488 Ki = 0.036 nM T50594 C06VMT 71624600 Ki = 0.009 nM T50594 CRP0B1 71624601 Ki = 0.061 nM T50594 CEA49N 71624602 Ki = 0.038 nM T50594 CG16LA 71624603 Ki = 0.015 nM T50594 C7AOZ0 71624604 Ki = 0.04 nM T50594 C7L6CY 71624710 Ki = 0.074 nM T50594 CQ8AR2 71624711 Ki = 0.025 nM T50594 CEFO84 71624712 Ki = 0.016 nM T50594 CWK48Z 71624713 Ki = 0.007 nM T50594 CY52PM 71624822 Ki = 0.007 nM T50594 CHW1F2 71723297 IC50 = 400 nM T50594 C4O8YU 71723298 IC50 = 220 nM T50594 COW25I 71723443 IC50 = 40 nM T50594 C97DCN 71723444 IC50 = 150 nM T50594 CCM0S5 71723445 IC50 = 200 nM T50594 CPG8H5 71723448 IC50 = 1100 nM T50594 CGY4Z5 71730239 IC50 = 0.4 nM T50594 CS2RT7 71730241 IC50 = 0.7 nM T50594 CEZ0Y3 71730242 IC50 = 1.6 nM T50594 CR80EU 71730367 IC50 = 1.2 nM T50594 C09BGX 71731146 IC50 = 0.8 nM T50594 C5ES1L 71731394 IC50 = 3 nM T50594 CC2UI1 71731515 IC50 = 0.3 nM T50594 C87XSZ 71731781 IC50 = 0.1 nM T50594 C8VPO2 71731919 IC50 = 2.6 nM T50594 CCQ3M7 72545499 IC50 = 1527 nM T50594 C4O9NE 72545500 IC50 = 804 nM T50594 CJ02UF 72545501 IC50 = 718 nM T50594 CCGY76 72545755 IC50 = 3.1 nM T50594 CET5H3 72545756 IC50 = 2.9 nM T50594 CK1IP9 72545757 IC50 = 6.8 nM T50594 CZ94IO 72545758 IC50 = 1.5 nM T50594 CGH65P 72545759 IC50 = 25 nM T50594 C9I7FZ 72545760 IC50 = 1618 nM T50594 CZ1P8N 72545761 IC50 = 5.1 nM T50594 C78DLB 72545995 IC50 = 5 nM T50594 C4TWP5 72545996 IC50 = 1.6 nM T50594 CV0T5B 72545997 IC50 = 2 nM T50594 CES3X4 72545998 IC50 = 7 nM T50594 CED7S2 72545999 IC50 = 7.2 nM T50594 CQG0D7 72546000 IC50 = 9.4 nM T50594 CBU13H 72546001 IC50 = 247 nM T50594 CJH0D1 72546229 IC50 = 10 nM T50594 C6CNJ9 72546230 IC50 = 834 nM T50594 CN43BE 72546231 IC50 = 3511 nM T50594 CL0F6B 72546232 IC50 = 4.5 nM T50594 C9E4XZ 72546233 IC50 = 1.3 nM T50594 CFZS35 72546235 IC50 = 136 nM T50594 CB0W2Y 72546472 IC50 = 162 nM T50594 CL03TU 72546473 IC50 = 834 nM T50594 C6OP8A 72696512 IC50 = 2544 nM T50594 C5DTG3 72696513 IC50 = 5471 nM T50594 C8ZGP7 72696514 IC50 = 2548 nM T50594 CKH1L5 72696643 IC50 = 1716 nM T50594 C3W0PQ 72696644 IC50 = 1937 nM T50594 CV3DQ2 72696645 IC50 = 521 nM T50594 CF23PI 72696646 IC50 = 1275 nM T50594 CVL7Y4 72696647 IC50 > 10000 nM T50594 CW3C1O 72696648 IC50 = 614 nM T50594 CFWX79 72696775 IC50 = 375 nM T50594 CA21RI 72696776 IC50 = 124 nM T50594 C4O7BN 72696777 IC50 = 94 nM T50594 CIWC01 72696778 IC50 = 33 nM T50594 CE1VB4 72696779 IC50 = 1098 nM T50594 C83EPX 72696908 IC50 = 125 nM T50594 CY0DG1 72696909 IC50 = 132 nM T50594 CL4RD1 72696910 IC50 > 5000 nM T50594 C1A6VK 72696912 IC50 = 13 nM T50594 CY5AR8 72696914 IC50 = 150 nM T50594 C49GBP 72696916 IC50 = 10 nM T50594 C4GLH1 72697053 IC50 = 16 nM T50594 CJEC10 72697054 IC50 = 87 nM T50594 CC1H2R 72697055 IC50 = 141 nM T50594 CUCG27 72697056 IC50 = 12 nM T50594 C1HB3Q 72697057 IC50 = 233 nM T50594 C1LOH7 72697202 IC50 = 2 nM T50594 C62JGC 72715291 Ki = 0.02 nM T50594 C6H7QA 72725546 Ki = 59 nM T50594 CJ15KC 72725547 Ki = 61 nM T50594 CQ5K4U 72725607 Ki = 4 nM T50594 C6SDB7 72737202 IC50 > 10000 nM T50594 CVF34X 73056835 IC50 = 0.3 nM T50594 CVY2Z3 73056836 IC50 = 1 nM T50594 C25CJV 73057145 IC50 = 0.4 nM T50594 CYLK14 73333219 IC50 = 130 nM T50594 CA51GV 73347322 IC50 = 1000 nM T50594 CHZ9U3 73352003 Ki = 0.057 nM T50594 C8MZG3 73354147 IC50 = 7 nM T50594 CXZ9J0 73356528 Ki = 0.011 nM T50594 CVF5P0 73603034 Ki = 0.03 nM T50594 C3UC9H 73891099 IC50 = 3100 nM T50594 CU5K6Q 74983184 Ki = 0.05 nM T50594 CVA40O 74983298 Ki = 0.003 nM T50594 C7R8WN 75364199 IC50 = 6.7 nM T50594 CK91CM 75365170 IC50 = 55 nM T50594 CYRP53 76310130 Ki > 12500 nM T50594 CV8QX0 76310169 IC50 > 30000 nM T50594 C49LJQ 76317357 Ki > 12500 nM T50594 CXZ30Q 76321071 Ki > 12500 nM T50594 CA5L4W 76324771 IC50 > 30000 nM T50594 C9GO0P 76328313 IC50 = 21300 nM T50594 CX4KN2 76331961 Ki = 460 nM T50594 CXG04C 76331962 Ki = 3300 nM T50594 CJER97 76331963 Ki = 2300 nM T50594 C0AYU9 76335538 Ki = 1000 nM T50594 C28YJW 76335539 Ki = 12300 nM T50594 C39FTZ 76335685 IC50 > 100000 nM T50594 C24USN 77050662 Ki = 0.018 nM T50594 CROJ27 78103829 Ki = 0.01 nM T50594 CGDC06 86294715 IC50 = 3 nM T50594 C3AF2E 86676680 Ki = 1300 nM T50594 C30ZNQ 86681992 IC50 = 2 nM T50594 CB7OC1 86681995 IC50 = 1.3 nM T50594 C5C1PH 86681998 IC50 = 3.8 nM T50594 C15JBI 86713879 Ki = 0.006 nM T50594 CK8V3O 86725098 IC50 = 312 nM T50594 C5R4CY 87057584 IC50 = 17 nM T50594 C4GF2R 89157636 IC50 = 25 nM T50594 C1HW4B 89735655 IC50 = 1600 nM T50594 CI57QV 89782019 IC50 = 0.34 nM T50594 CAG7B6 89782150 IC50 = 0.1 nM T50594 CH8JN1 89783250 IC50 = 0.2 nM T50594 C1CL8I 89783341 IC50 = 0.1 nM T50594 CUNJ79 89783434 IC50 = 0.6 nM T50594 CRQM10 89783564 IC50 = 5 nM T50594 CPX3K8 89783643 IC50 = 0.17 nM T50594 C2K3DA 89783801 IC50 = 0.2 nM T50594 CPQ9L3 89783993 IC50 = 0.9 nM T50594 C16ZQO 89784003 IC50 = 0.5 nM T50594 CDCO54 89784354 IC50 = 3 nM T50594 C8X1VA 89784686 IC50 = 0.07 nM T50594 CX2H4B 89784954 IC50 = 6.6 nM T50594 C0JIS8 89793954 IC50 = 44 nM T50594 C3N2TQ 89914568 Ki = 0.07 nM T50594 CXF3T0 90058666 IC50 = 0.1 nM T50594 C1UJ8Q 90058675 IC50 = 0.4 nM T50594 CWRJ32 90058676 IC50 = 1 nM T50594 CYZ98S 90058679 IC50 = 0.6 nM T50594 CFH4L6 90058683 IC50 = 0.07 nM T50594 CV9KG7 90058690 IC50 = 0.3 nM T50594 CP13IU 90058693 IC50 = 1 nM T50594 C56AJL 90058786 IC50 = 2 nM T50594 C35WJR 90058791 IC50 = 0.06 nM T50594 CCA78J 90058814 IC50 = 0.1 nM T50594 CN6H2I 90058905 IC50 = 0.5 nM T50594 C7DVW3 90058906 IC50 = 0.3 nM T50594 CCSB80 90072314 Ki = 0.006 nM T50594 C1J4AE 90072384 Ki = 0.01 nM T50594 CW4YI5 90072542 Ki = 0.003 nM T50594 CR34AN 90073003 Ki = 0.071 nM T50594 CYW61R 90256619 IC50 = 2 nM T50594 CK79BW 90256983 IC50 = 11 nM T50594 CX8NV6 90257109 IC50 = 262 nM T50594 CX4J8N 90286701 IC50 = 1000 nM T50594 C75FLG 90326903 IC50 = 0.021 nM T50594 CN0V6L 90326906 IC50 = 0.037 nM T50594 CY0UC4 90645194 IC50 = 1441 nM T50594 CEV5P2 90645195 IC50 = 838 nM T50594 C3E6PB 90656756 IC50 = 45.1 nM T50594 C95SGV 90656757 IC50 = 20.4 nM T50594 C0MWE6 90656758 IC50 = 25.8 nM T50594 CR3J7I 90656759 IC50 = 18.7 nM T50594 CHK6P8 90656760 IC50 = 34.5 nM T50594 CI68DP 90656761 IC50 = 2.8 nM T50594 COC3M0 90656762 IC50 = 18.3 nM T50594 C7JM5Z 90656763 IC50 = 17.2 nM T50594 C3MQ1Z 90656764 IC50 = 8 nM T50594 CL0AN8 90656765 IC50 = 1130 nM T50594 C7B9YM 90656766 IC50 = 370 nM T50594 C84CTN 90656767 IC50 = 270 nM T50594 C62DBJ 90656768 IC50 = 270 nM T50594 C1WQT0 90656769 IC50 = 400 nM T50594 C7L8SK 95040885 IC50 = 25 nM T50594 C10XIT 101898720 IC50 = 70 nM T50594 C5N1VZ 102581295 IC50 > 10000 nM T50594 CJ7XB9 118711716 IC50 = 120 nM T50594 C0A2RY 118720249 IC50 = 1 nM T50594 C95FJY 118720250 IC50 = 34 nM T50594 C06XZY 118720251 IC50 = 550 nM T50594 CVK71Z 118720252 IC50 = 49 nM T50594 C3CB8J 118720253 IC50 = 21 nM T50594 CV3ZY2 118720254 IC50 = 5000 nM T50594 CNI0U1 118720255 IC50 = 21 nM T50594 CIX9N3 118720917 IC50 = 633 nM T50594 CH09OX 118720918 IC50 = 149 nM T50594 CVM73U 118721227 IC50 = 186 nM T50594 CXY1K0 118721228 IC50 = 168 nM T50594 CEHY81 118725601 IC50 = 3 nM T50594 C6J7VS 118725602 IC50 = 3 nM T50594 CRY0X4 118725603 IC50 = 25 nM T50594 CY4P9O 118725604 IC50 = 0.9 nM T50594 CAT0C1 118725605 IC50 = 1.6 nM T50594 CL6CM1 118725606 IC50 = 4 nM T50594 C6JNB7 118725607 IC50 = 2 nM T50594 CE3B5A 118725608 IC50 = 4 nM T50594 C36FLX 118725609 IC50 = 3 nM T50594 CG6I4T 118725610 IC50 = 3 nM T50594 CN82QT 118725611 IC50 = 0.2 nM T50594 CUN73P 118725613 IC50 = 0.5 nM T50594 CL5K0U 118725614 IC50 = 1.4 nM T50594 CXEP50 118725615 IC50 = 0.3 nM T50594 CTUD48 118725865 IC50 = 2830 nM T50594 CQCX41 118737057 IC50 > 10000 nM T50594 C4X7SD 122192466 IC50 = 4037 nM T50594 C0NE4L 122193063 IC50 = 42 nM T50594 CC7WL9 122193064 IC50 = 9 nM T50594 CZ1NE6 122194258 IC50 = 1400 nM T50594 CO3K9M 122194259 IC50 = 1560 nM T50594 CI1N4B 122194260 IC50 = 390 nM T50594 CS86FI 122194261 IC50 = 1100 nM T50594 C4V5AG 122194268 IC50 = 740 nM T50594 C5EH2L 122196349 Ki = 8.5 nM T50594 CKR45A 122196350 Ki = 0.02 nM T50594 CIF59P 122196351 Ki = 3.4 nM T50594 C2ES7U 122196352 Ki = 800 nM T50594 C4I2VM 122196353 Ki = 3200 nM T50594 CBW2O1 122373914 IC50 = 10600 nM T50594 CZD9W8 123518123 IC50 = 20 nM T50594 C0T6VF 123561371 IC50 = 7 nM T50594 C04QEN 123616291 Ki = 0.03 nM T50594 C7G6IA 123944769 IC50 = 18 nM T50594 CDL2V4 124005596 EC50 = 283 nM T50594 C7PN8C 127028369 IC50 > 10000 nM T50594 C5S2BD 127028699 IC50 = 1050 nM T50594 C8EBD3 127028700 IC50 = 1870 nM T50594 C6C1MY 127028701 IC50 > 10000 nM T50594 C24FSM 127028702 IC50 = 800 nM T50594 CG52VH 127029004 IC50 = 2470 nM T50594 C8TLM3 127029011 IC50 = 2100 nM T50594 C1GCY3 127029012 IC50 = 2020 nM T50594 CI8V6G 127029013 IC50 > 10000 nM T50594 C0HN2Y 127030123 IC50 = 16410 nM T50594 C7S9GI 127030124 IC50 > 100000 nM T50594 CHGN68 127030424 IC50 = 2810 nM T50594 CRV62L 127030425 IC50 > 100000 nM T50594 CF7JT8 127030426 IC50 > 100000 nM T50594 C5YCU2 127030427 IC50 > 100000 nM T50594 CRA5S2 127030832 IC50 = 750 nM T50594 C0GES2 127031075 IC50 > 100000 nM T50594 CFJ32Y 127031076 IC50 > 100000 nM T50594 CC8V4J 127031368 IC50 > 100000 nM T50594 C78GYH 127031383 IC50 > 100000 nM T50594 C5WA9Z 127031384 IC50 > 100000 nM T50594 CD7LN1 127031385 IC50 = 4910 nM T50594 CI0VX4 127031386 IC50 > 100000 nM T50594 CO89TC 127031387 IC50 = 11800 nM T50594 CAM4S5 127031675 IC50 > 100000 nM T50594 C4QD0M 127031676 IC50 = 27400 nM T50594 C0LTC3 127031677 IC50 > 100000 nM T50594 C4ZS6N 127032072 Ki < 1 nM T50594 CO1G2K 127032542 IC50 > 100000 nM T50594 C12IOL 127033165 IC50 > 100000 nM T50594 C5RO0L 127033758 IC50 > 100000 nM T50594 CRQ2J3 127033854 IC50 > 10000 nM T50594 CD04YX 127034308 IC50 > 31600 nM T50594 CS93KM 127037885 IC50 = 1080 nM T50594 CC05GQ 127037886 IC50 > 10000 nM T50594 C7F3JO 127038195 IC50 = 1450 nM T50594 CB5EU1 127038203 IC50 = 1310 nM T50594 CJI5T2 127039244 IC50 = 2040 nM T50594 CD4FK5 127039245 IC50 = 600 nM T50594 CDYA59 127039857 IC50 = 690 nM T50594 C1G4ES 127041542 Ki < 1 nM T50594 C8K0WU 127042183 Ki < 1 nM T50594 C94CGA 127042762 IC50 > 10000 nM T50594 CB4I2Y 127043000 IC50 = 27000 nM T50594 CU95YJ 127050291 IC50 = 150 nM T50594 CFKY32 129012056 IC50 = 250 nM T50594 CP16OG 129795093 IC50 = 1341 nM T50594 C46KZG 131704449 IC50 = 2500 nM T50594 CCPZ70 131704452 IC50 = 900 nM T50594 C4Q5LF 132471857 IC50 = 120 nM T50594 C8PLI9 132486774 IC50 = 54871000 nM T50594 CI8N3T 132486776 IC50 = 56511000 nM T50594 CIN9H0 132486780 IC50 = 3387 nM T50594 C0K5XP 132942309 IC50 = 2.2 nM T50594 C39UCD 133080605 IC50 = 43 nM T50594 C1W4DO 134135721 IC50 = 0.29 nM T50594 C9Z3XH 134138985 IC50 = 65 nM T50594 CX3A0W 134146922 IC50 = 0.04 nM T50594 C2AN7T 134611886 IC50 > 100000 nM T50594 CGBZ13 134843302 IC50 = 900 nM T50594 C4TED6 135418395 IC50 = 1700 nM T50594 C0A7EC 135428100 IC50 > 10000 nM T50594 CK73WQ 135430368 IC50 = 2100 nM T50594 C6AZ2R 135435018 IC50 = 501.19 nM T50594 C8KU4A 135436186 IC50 > 10000 nM T50594 C2O0WH 135439519 IC50 = 700 nM T50594 CSNE45 135461314 IC50 = 526 nM T50594 C7KI2H 135494325 IC50 = 3100 nM T50594 CK3NO2 135501994 IC50 = 184 nM T50594 CJXW63 135508850 IC50 = 2000 nM T50594 C2H7SQ 135508851 IC50 = 2500 nM T50594 C8B0YI 135513898 IC50 = 500 nM T50594 C4I1LU 135542186 IC50 = 5500 nM T50594 C2UO7P 135566502 Ki = 1 nM T50594 CFN90Y 135566503 Ki = 5 nM T50594 CY4D8I 135566504 Ki = 130.1 nM T50594 C5DOH6 135566645 IC50 = 17 nM T50594 CN4T8V 135566646 IC50 = 7 nM T50594 CN6E1U 135566647 IC50 = 27 nM T50594 CH2YR7 135566648 IC50 = 11 nM T50594 C5ILD8 135589827 IC50 = 75 nM T50594 CN2B3D 135747628 IC50 = 0.05 nM T50594 CA6EQ3 135856841 Ki = 5 nM T50594 CO32WX 135856854 Ki = 14 nM T50594 C4X7QD 135856859 Ki = 12 nM T50594 C78FMI 135856860 Ki = 332 nM T50594 CCJR27 135856881 Ki = 44 nM T50594 C1CN9W 135856896 Ki = 42 nM T50594 CPL2Q0 135856897 Ki = 11 nM T50594 CLYW16 135856902 Ki = 5 nM T50594 CR8S9H 135856912 Ki = 71 nM T50594 CO47YW 135856913 Ki = 17 nM T50594 C39TEH 135856921 Ki = 11 nM T50594 C1KP2E 135860183 IC50 = 3100 nM T50594 CK9M5H 135867902 IC50 = 16 nM T50594 C20HYR 135867903 IC50 = 24 nM T50594 CZ70TA 135867906 IC50 = 14 nM T50594 C0MSR4 135867912 IC50 = 35 nM T50594 CGM17H 135867918 IC50 = 61 nM T50594 CUQ51Z 135867923 IC50 = 28 nM T50594 C0J7RQ 135867925 IC50 = 640 nM T50594 CORN45 135867927 IC50 = 580 nM T50594 C9JBD1 135867931 IC50 = 142 nM T50594 CEX54P 135867940 IC50 = 6 nM T50594 C4XA7O 135867941 IC50 = 3.8 nM T50594 C8MR6U 135867952 IC50 = 5000 nM T50594 C0M9LS 135867953 IC50 = 23 nM T50594 CP1VS6 135867954 IC50 = 376 nM T50594 CIV27R 135867956 IC50 = 497 nM T50594 CN8PW9 135867959 IC50 = 1871 nM T50594 CWSI79 135867966 IC50 = 232 nM T50594 CTPK14 135867967 IC50 = 205 nM T50594 CXU39R 135867972 IC50 = 99 nM T50594 C2CZ9L 135867976 IC50 = 15 nM T50594 C7JP3T 135867977 IC50 = 73 nM T50594 CDYQ36 135867981 IC50 = 32 nM T50594 CP56XU 135867984 IC50 = 77 nM T50594 C28JUY 135867996 IC50 = 3963 nM T50594 C1GBJ8 135867997 IC50 = 8 nM T50594 CC92BK 135867998 IC50 = 11 nM T50594 C6RU2Z 135868002 IC50 = 281 nM T50594 CGX7J5 135885107 IC50 = 6200 nM T50594 CMF2T3 135909509 IC50 = 1770 nM T50594 CK2EH9 135921041 Ki = 0.8 nM T50594 C02PHA 135927892 IC50 = 316.23 nM T50594 CS8T3D 135927897 IC50 = 125.89 nM T50594 CW0XS9 135927905 Ki = 16 nM T50594 CB0X1D 135927906 Ki = 296 nM T50594 C97XNC 135927907 Ki = 33 nM T50594 CCEL26 135927908 Ki = 0.9 nM T50594 C3G8VW 135927909 Ki = 92 nM T50594 C3YD9J 135927910 Ki = 18 nM T50594 CS9VK5 135927911 Ki = 32 nM T50594 CZ53AS 135927912 Ki = 36 nM T50594 CEI85B 135927919 Ki = 11 nM T50594 CB5N8A 135927920 Ki = 65 nM T50594 CCV12A 135927921 Ki = 3 nM T50594 C42TUA 135927922 Ki = 14 nM T50594 C1AJ7H 135927923 Ki = 5 nM T50594 CGUR31 135927924 Ki = 2 nM T50594 CG34TQ 135927925 Ki = 4 nM T50594 CIW7F3 135927928 Ki = 4 nM T50594 CX1B7W 135927929 Ki = 11 nM T50594 CWX70K 135927931 Ki = 9 nM T50594 C7HER4 135927932 Ki = 92 nM T50594 CXOE95 135927933 Ki = 107 nM T50594 CZOK96 135927935 Ki = 3 nM T50594 C34ZBN 135927936 Ki = 66 nM T50594 C47RLS 135927937 Ki = 38 nM T50594 CV3H7I 135927938 Ki = 49 nM T50594 C19LMJ 135927939 Ki = 20 nM T50594 CZ25EG 135927940 Ki = 9 nM T50594 C4M7IK 135927941 Ki = 5 nM T50594 CX9SA7 135927946 Ki = 4 nM T50594 C90WDM 135927947 Ki = 6 nM T50594 C7E1TR 135927948 Ki = 5 nM T50594 CEXC86 135927949 Ki = 1 nM T50594 COM4E6 135927950 Ki = 5 nM T50594 C3QTI7 135927951 Ki = 12 nM T50594 CKN37Q 135927952 Ki = 1 nM T50594 C7RLI0 135927958 Ki = 40 nM T50594 CK8Z5W 135927959 Ki = 8 nM T50594 CCX4E5 135927960 Ki = 4 nM T50594 C0ZP1O 135927961 Ki = 8 nM T50594 CP6W0X 135927962 Ki = 8 nM T50594 CPX81K 135927963 Ki = 2 nM T50594 C6F1QB 135927964 Ki = 29 nM T50594 CH1I0A 135927969 Ki = 1 nM T50594 C36KIX 135927970 Ki = 0.6 nM T50594 C28JYO 135927971 Ki = 2 nM T50594 C35IDA 135927972 Ki = 2 nM T50594 CN0J8C 135927973 Ki = 3 nM T50594 CG3UZ1 135927974 Ki = 0.7 nM T50594 C5E2KU 135927977 Ki = 271 nM T50594 C2OJK4 135927978 Ki = 4 nM T50594 C14JUY 135927979 Ki = 0.8 nM T50594 C1H2EG 135927980 Ki = 43 nM T50594 C7ZD2B 135928468 Ki = 3 nM T50594 C14OBQ 135928469 Ki = 2 nM T50594 C7C3MX 135928470 Ki = 4 nM T50594 CYTA89 135930672 IC50 = 13 nM T50594 CZWV36 135961524 IC50 = 130 nM T50594 CHA4N2 136013680 IC50 > 10 nM T50594 CR1P5M 136025848 IC50 = 4600 nM T50594 CG39ZH 136025849 IC50 = 6100 nM T50594 C85XKB 136025991 IC50 = 3500 nM T50594 C7P0NV 136025992 IC50 > 10000 nM T50594 CC4UG2 136025994 IC50 = 5000 nM T50594 C63KRL 136026134 IC50 > 10000 nM T50594 C2OP5Y 136026135 IC50 > 10000 nM T50594 CKL49A 136026136 IC50 = 2500 nM T50594 C1HV2M 136026137 IC50 = 1500 nM T50594 CTX08I 136026138 IC50 = 4500 nM T50594 CBO76R 136026139 IC50 = 2100 nM T50594 C8QU9L 136026140 IC50 = 6500 nM T50594 C7OKA9 136033523 IC50 = 2000 nM T50594 CV0U7E 136033524 IC50 = 4200 nM T50594 CHQO83 136033525 IC50 = 2100 nM T50594 CO34IK 136033527 IC50 = 300 nM T50594 CQS9R7 136033528 IC50 > 10000 nM T50594 CD1A7S 136033529 IC50 = 3700 nM T50594 C6VH4F 136033539 IC50 > 10000 nM T50594 C4H9ZD 136033543 IC50 > 10000 nM T50594 CC54MD 136033544 IC50 = 3100 nM T50594 C2AO3G 136033545 IC50 = 9000 nM T50594 CJ98EN 136033546 IC50 = 1200 nM T50594 C3I7UD 136033547 IC50 > 10000 nM T50594 CVFW17 136033548 IC50 > 10000 nM T50594 C3YL4I 136042193 IC50 = 2 nM T50594 CAW0E4 136065882 IC50 > 100000 nM T50594 CSV8T4 136068690 IC50 > 10000 nM T50594 CP7H8T 136086742 IC50 > 10000 nM T50594 CSNQ71 136086752 IC50 = 7000 nM T50594 CI19RB 136086756 IC50 = 4500 nM T50594 C98FHO 136086762 IC50 = 2800 nM T50594 CCVU40 136086892 IC50 = 7200 nM T50594 CHR1T4 136086893 IC50 = 4000 nM T50594 CM84LZ 136086894 IC50 > 10000 nM T50594 C13DGL 136086895 IC50 = 590 nM T50594 COV8E0 136094762 IC50 = 28000 nM T50594 CS4R2M 136098630 IC50 = 9 nM T50594 CWM2S3 136098631 IC50 = 30 nM T50594 CL1NA0 136109067 IC50 > 10000 nM T50594 CCB70U 136123533 Ki = 358 nM T50594 CP3CA4 136189660 IC50 = 3 nM T50594 CQY0C7 136189673 IC50 = 18 nM T50594 CC52HL 136189674 IC50 = 5 nM T50594 C4G9BI 136189695 IC50 = 9 nM T50594 CC87DY 136189770 IC50 = 2982 nM T50594 CQGO78 136189786 IC50 = 77 nM T50594 CTL8M5 136189797 IC50 = 3 nM T50594 C5N2QZ 136189800 IC50 = 22 nM T50594 CC40LU 136189802 IC50 = 39 nM T50594 CX45QN 136189847 IC50 = 24 nM T50594 CO8B4N 136189863 IC50 = 11 nM T50594 CJ57SF 136189870 IC50 = 102 nM T50594 CTVX09 136189895 IC50 = 4 nM T50594 CFZT23 136189934 IC50 = 4 nM T50594 CB6EY8 136189986 IC50 = 65 nM T50594 CCWV39 136189998 IC50 = 72 nM T50594 C9SP0D 136190004 IC50 = 77 nM T50594 CZ1DH2 136190005 IC50 = 104 nM T50594 CYR45B 136190013 IC50 = 31 nM T50594 CV9N1O 136190017 IC50 = 10 nM T50594 CJ5LB9 136190029 IC50 = 46 nM T50594 CQ85IN 136190059 IC50 = 18 nM T50594 CX8TS5 136190062 IC50 = 10 nM T50594 CU0MZ9 136190070 IC50 = 11 nM T50594 CLW25G 136190081 IC50 = 293 nM T50594 C1YUD0 136219394 IC50 > 10 nM T50594 CAY7U9 136236280 IC50 = 3 nM T50594 C73IGY 136244208 IC50 = 7 nM T50594 CXS5Z6 136254223 IC50 = 5000 nM T50594 C2DNM5 136254224 IC50 > 5000 nM T50594 CQM1U4 136254225 IC50 = 3 nM T50594 COU4C5 136254226 IC50 = 5000 nM T50594 CQU6J7 136254227 IC50 = 5000 nM T50594 CIU8W3 136254389 IC50 > 10 nM T50594 CL95WA 136380901 IC50 = 1.9 nM T50594 C3MK9W 136807986 IC50 > 10000 nM T50594 C4VAQ0 136966273 IC50 = 0.4 nM T50594 CVG90R 137631416 IC50 = 1 nM T50594 CYEV23 137632380 IC50 = 8 nM T50594 CYQJ28 137632388 IC50 = 8 nM T50594 CY37WA 137632732 IC50 = 36 nM T50594 CPQ6V8 137633459 IC50 = 36 nM T50594 CV1A5N 137633544 IC50 = 23 nM T50594 C8T1DE 137634063 IC50 = 156 nM T50594 CI1E8V 137634241 IC50 > 10000 nM T50594 CC9DG4 137634486 IC50 = 1.4 nM T50594 C6D8IM 137634495 IC50 = 43 nM T50594 CK7QM8 137634713 Ki = 190 nM T50594 CXGL06 137634918 IC50 = 70 nM T50594 C9AIT8 137634969 IC50 = 0.64 nM T50594 CJ65FX 137635465 IC50 = 624 nM T50594 C0BYO6 137635499 IC50 = 2 nM T50594 CS27HQ 137635523 IC50 = 25500 nM T50594 CN34DS 137635572 IC50 = 16 nM T50594 C05LXW 137635643 IC50 = 100 nM T50594 CK52BV 137635684 IC50 = 2.4 nM T50594 C8D7TE 137635945 IC50 = 554 nM T50594 CA1D9B 137636162 IC50 = 31 nM T50594 CF65JZ 137636187 IC50 = 0.41 nM T50594 CD5IZ6 137636389 Ki = 0.5 nM T50594 CSQ0T2 137636417 IC50 = 1 nM T50594 CQ5S9H 137636735 IC50 = 3 nM T50594 CK3OH2 137636993 IC50 = 7 nM T50594 CU9YQ3 137637635 IC50 = 1790 nM T50594 C5HD0W 137638179 IC50 = 1 nM T50594 C3GTQ2 137638400 IC50 = 335 nM T50594 C1MO4H 137638461 IC50 = 2 nM T50594 CUF1D9 137638752 Ki = 0.5 nM T50594 C21XCP 137638981 IC50 = 4 nM T50594 CJ69GR 137638996 IC50 = 4 nM T50594 CX1O0W 137639052 IC50 = 273 nM T50594 CU8R7Z 137639370 IC50 = 332 nM T50594 C6SE7H 137639744 IC50 = 775 nM T50594 CWR2B4 137640402 IC50 = 784 nM T50594 CV5M4H 137640638 IC50 = 1.1 nM T50594 C25JLY 137640893 IC50 = 31 nM T50594 CO2WM4 137640946 IC50 = 2.1 nM T50594 CL9Y0K 137640988 IC50 = 4 nM T50594 C9EBK4 137641161 IC50 = 6.8 nM T50594 CI0NF6 137641367 IC50 > 30000 nM T50594 C1TFP0 137641562 IC50 = 2 nM T50594 C60YZT 137641798 IC50 = 49 nM T50594 C8FOH1 137642030 IC50 = 2 nM T50594 CS9HF4 137642256 IC50 = 4800 nM T50594 C30DWC 137642509 Ki = 38 nM T50594 CO03XB 137642855 IC50 = 2 nM T50594 CPO2G4 137642902 IC50 = 8 nM T50594 CHD90A 137643257 Ki = 0.8 nM T50594 C2MO5L 137643556 IC50 = 12 nM T50594 CHOI53 137643582 IC50 = 4 nM T50594 CNL3U7 137643747 IC50 = 42 nM T50594 CL6K4E 137643873 IC50 = 28 nM T50594 CE8GA3 137644163 IC50 = 25 nM T50594 CJS20N 137644367 IC50 = 3 nM T50594 C0DAH4 137644542 IC50 = 32 nM T50594 CDA2N6 137644922 IC50 = 77 nM T50594 C2ZXK8 137645147 IC50 = 0.28 nM T50594 CGB8T4 137645179 IC50 = 1030 nM T50594 CY23WH 137645765 IC50 = 267 nM T50594 C2D9SE 137645829 IC50 = 5 nM T50594 CB2Z5V 137646513 IC50 = 37 nM T50594 C1H3ZK 137647783 IC50 = 1 nM T50594 C3JDR6 137648580 Ki = 0.7 nM T50594 C7UTE8 137648598 IC50 = 1 nM T50594 CD08UY 137648872 IC50 = 974 nM T50594 CVP1A8 137649309 IC50 = 127 nM T50594 CCF3T5 137649330 IC50 = 9.2 nM T50594 C93ANB 137649688 IC50 = 16 nM T50594 CL2J6B 137649761 IC50 = 171 nM T50594 CZ37HC 137649765 IC50 = 295 nM T50594 CBWI50 137649962 IC50 = 11 nM T50594 CCZE58 137650076 IC50 = 67 nM T50594 CAK39E 137650557 IC50 = 250 nM T50594 CDF3Q7 137650805 IC50 = 250 nM T50594 C8J3RF 137651484 IC50 = 2 nM T50594 CEDP85 137651503 IC50 = 3335 nM T50594 C8AYS0 137651935 IC50 = 85 nM T50594 CBA35I 137652021 IC50 = 19250 nM T50594 CYGH52 137652180 IC50 = 940 nM T50594 C7SB9W 137652377 IC50 = 1200 nM T50594 C2EA4F 137652505 IC50 = 3 nM T50594 CIHD74 137653335 IC50 = 10040 nM T50594 C0U7AR 137653670 IC50 = 804 nM T50594 C6JZ8E 137654438 IC50 = 1.8 nM T50594 C4CWB2 137654577 IC50 = 8 nM T50594 C35CMU 137654615 IC50 = 3.6 nM T50594 CIZ8M6 137654684 IC50 = 13 nM T50594 CSQG93 137654724 IC50 = 1 nM T50594 C2UV8N 137654823 IC50 = 1160 nM T50594 CB5A0K 137655276 IC50 = 131 nM T50594 CZE82A 137655925 IC50 = 1 nM T50594 C2T0KO 137655995 IC50 = 68 nM T50594 CFXC14 137656007 Ki = 0.02 nM T50594 C7AYN9 137656129 IC50 = 4.5 nM T50594 C1BEV7 137656991 IC50 = 6 nM T50594 CD60ZK 137657358 IC50 = 2.9 nM T50594 C3VL2F 137657596 IC50 = 10000 nM T50594 C3H9BS 137657667 IC50 = 2 nM T50594 CR9F6C 137657836 IC50 = 2 nM T50594 CU6Q4J 137658394 IC50 = 1470 nM T50594 CZRW59 137659000 IC50 = 304 nM T50594 CTC53Y 137659105 IC50 = 16 nM T50594 CF25MB 137659327 IC50 = 0.7 nM T50594 C72ZDI 137659673 Ki = 0.4 nM T50594 C70GPH 137659881 IC50 = 103 nM T50594 CK03MR 137660117 IC50 = 720 nM T50594 C4OUD0 137660252 Ki = 450 nM T50594 C92YUI 137660945 IC50 = 107 nM T50594 C1XVG6 137661399 IC50 = 175 nM T50594 CUK0R8 137661493 IC50 = 2124 nM T50594 CW57TM 137661945 IC50 = 125 nM T50594 CQ82UE 137662204 IC50 = 1000 nM T50594 C7N3ZQ 145951035 IC50 = 2800 nM T50594 CML51F 145951743 IC50 = 1010 nM T50594 C0T5JZ 145952083 IC50 > 10000 nM T50594 C1W0GJ 145952796 IC50 = 15848.93 nM T50594 CL47SB 145953112 IC50 > 10000 nM T50594 C80DPI 145953422 IC50 > 10000 nM T50594 CEV70S 145953574 IC50 = 760 nM T50594 CQ35PD 145954426 IC50 > 10000 nM T50594 CIR3O7 145955130 IC50 > 10000 nM T50594 CG6D7S 145955812 IC50 > 10000 nM T50594 CEG10W 145955965 IC50 > 10000 nM T50594 CC1Z6W 145956369 IC50 > 10000 nM T50594 CWNX41 145957259 IC50 > 10000 nM T50594 CMJ5D9 145958016 IC50 = 290 nM T50594 CUD58Z 145959186 IC50 > 10000 nM T50594 CT30CG 145960449 IC50 = 1290 nM T50594 CS32YP 145960484 IC50 = 21 nM T50594 CE9D6T 145960511 IC50 > 10000 nM T50594 CHZ20V 145960670 IC50 = 257 nM T50594 C81DKZ 145960765 IC50 = 7 nM T50594 C8M2RY 145960938 IC50 = 30 nM T50594 CNSO87 145961054 IC50 = 12 nM T50594 CD2O0Q 145961184 IC50 = 8 nM T50594 CY25XU 145961279 IC50 = 9 nM T50594 C8IAB5 145961349 IC50 = 21 nM T50594 CDTI85 145961440 IC50 = 19 nM T50594 CXU40G 145961470 IC50 = 5 nM T50594 CW15YM 145961475 IC50 = 307 nM T50594 CUI86V 145961560 IC50 = 260 nM T50594 CE26LP 145961625 IC50 = 160 nM T50594 CV15YW 145961659 IC50 = 5 nM T50594 C0KY1T 145961724 IC50 = 313 nM T50594 C2YQF0 145961914 IC50 = 35 nM T50594 CH2V4T 145961915 IC50 = 7 nM T50594 CQLA92 145961972 IC50 = 9 nM T50594 C4M6SJ 145961986 IC50 > 10000 nM T50594 COW23H 145962040 IC50 = 9 nM T50594 C7OF6V 145962094 IC50 = 3 nM T50594 CB3O4I 145962109 IC50 = 885 nM T50594 CP3EH0 145962188 IC50 = 9 nM T50594 C9S8AO 145962192 IC50 = 7 nM T50594 CZIT45 145962335 IC50 = 33 nM T50594 CTN2B1 145962545 IC50 = 144 nM T50594 C5NCH1 145962614 IC50 = 195 nM T50594 C2TRN8 145962743 IC50 = 256 nM T50594 CLS90K 145962852 IC50 = 134 nM T50594 CJD24A 145962897 IC50 = 22 nM T50594 C9C3YP 145962963 IC50 = 67 nM T50594 C69ZIQ 145963064 IC50 > 10000 nM T50594 C01JIP 145963077 IC50 = 443 nM T50594 CJQ78W 145963108 IC50 = 187 nM T50594 CY8RS4 145963277 IC50 = 96 nM T50594 CUI0L7 145963307 IC50 = 23 nM T50594 CO4Y1M 145963467 IC50 = 3 nM T50594 C8QDJ0 145963511 IC50 = 209 nM T50594 C1J5BC 145963517 IC50 = 21 nM T50594 C3TLW0 145963725 IC50 = 19 nM T50594 CNF4J3 145966584 IC50 = 58 nM T50594 CV28AL 145967603 IC50 = 5300 nM T50594 C5B0QL 145967935 IC50 = 830 nM T50594 CMG01Q 145968043 IC50 = 3400 nM T50594 C9LBY8 145968158 IC50 = 16800 nM T50594 CPET15 145968269 IC50 = 12000 nM T50594 C24AQX 145968504 IC50 > 30000 nM T50594 CTY0I5 145968604 IC50 = 14100 nM T50594 CL07SI 145968637 IC50 = 200 nM T50594 C7B3UD 145968656 IC50 = 630 nM T50594 CZN38I 145969224 IC50 > 30000 nM T50594 CL8V5N 145969695 IC50 > 30000 nM T50594 CAU16Y 145969796 IC50 = 2000 nM T50594 CISA20 145969798 IC50 > 30000 nM T50594 CM6D9P 145969896 IC50 = 2100 nM T50594 CT3N9K 145970124 IC50 = 1800 nM T50594 CQR9Z4 145970125 IC50 = 1200 nM T50594 CP0M6D 145970925 IC50 = 90 nM T50594 CQ4WO3 145971039 IC50 = 220 nM T50594 CD97BO 145971046 IC50 > 30000 nM T50594 C09DLU 145971051 IC50 = 3300 nM T50594 CX9PG6 145972012 IC50 = 74 nM T50594 C1JRY9 145972182 IC50 > 10000 nM T50594 CN42KR 145972228 IC50 > 10000 nM T50594 C07KNU 145977912 IC50 = 67 nM T50594 CVES49 145982552 IC50 > 10000 nM T50594 CIDU48 145982789 IC50 > 10000 nM T50594 CPO43Z 145982872 IC50 > 10000 nM T50594 CORV50 145982985 IC50 > 10000 nM T50594 C6YBK0 145983031 IC50 = 5000 nM T50594 CD3WR9 145983454 IC50 = 4500 nM T50594 CQXC48 145983553 IC50 > 10000 nM T50594 CJ4N1S 145983820 IC50 > 10000 nM T50594 C8GVD0 145984001 IC50 > 10000 nM T50594 CTJW32 145984202 IC50 > 10000 nM T50594 C48YNJ 145985058 IC50 > 10000 nM T50594 C67EVF 145985214 IC50 > 10000 nM T50594 CKQ69G 145985465 IC50 > 10000 nM T50594 C4P8SD 145989719 IC50 = 160 nM T50594 CYGN68 155510554 EC50 = 179 nM T50594 C25TBW 155511840 IC50 = 0.21 nM T50594 CC1V3X 155511863 IC50 = 0.06 nM T50594 CG7X2E 155512906 IC50 = 425 nM T50594 C2MD1Q 155513187 IC50 > 10000 nM T50594 CDF0I2 155514882 EC50 = 865 nM T50594 C7BMF4 155515543 IC50 = 0.09 nM T50594 C4RFU7 155516598 IC50 = 1.2 nM T50594 C4VKM8 155516837 IC50 = 785 nM T50594 CU35GB 155517528 IC50 = 5.8 nM T50594 CS3E7L 155518082 IC50 = 0.56 nM T50594 CY49NZ 155518625 IC50 = 2 nM T50594 C24NBM 155518799 IC50 = 0.08 nM T50594 C4T6CH 155518837 IC50 = 13 nM T50594 CO58XZ 155519799 Ki = 0.1 nM T50594 CKD52G 155520766 EC50 = 265 nM T50594 CJ5L2U 155520986 Ki = 0.2 nM T50594 CV42MB 155521123 IC50 = 0.03 nM T50594 CM8HF6 155521436 Ki = 0.04 nM T50594 CQ74ZC 155521929 IC50 = 870 nM T50594 CGQH30 155523583 Ki = 0.03 nM T50594 C5SWL6 155524053 IC50 > 10000 nM T50594 CUM08K 155524352 IC50 = 0.29 nM T50594 CQ0I3P 155524597 IC50 = 236 nM T50594 C3BTZ8 155525211 Ki = 0.08 nM T50594 CY7EM6 155525492 IC50 = 2.4 nM T50594 CX59UT 155526046 IC50 = 1.6 nM T50594 CE5ZU0 155526194 IC50 = 30 nM T50594 CQ4XA9 155527433 IC50 = 7 nM T50594 C5OBZ9 155527556 Ki = 0.007 nM T50594 C76QNG 155528354 EC50 = 322 nM T50594 CR5ON6 155528414 IC50 = 0.36 nM T50594 C2R8JO 155528784 IC50 = 420 nM T50594 CN0M8O 155529692 IC50 = 0.65 nM T50594 CEF14U 155529807 IC50 = 0.12 nM T50594 C5T4ZI 155530130 IC50 = 1100 nM T50594 CS9W1N 155531462 IC50 = 1.7 nM T50594 C2N6XM 155531935 IC50 = 17 nM T50594 CY59IV 155531989 IC50 = 2.3 nM T50594 C8IP7E 155532982 IC50 = 7 nM T50594 C3K2ZL 155533051 IC50 = 0.11 nM T50594 CIH5W7 155534088 IC50 = 0.14 nM T50594 C9SLQ4 155534205 IC50 = 111.01 nM T50594 CL7U8D 155534608 Ki = 1.2 nM T50594 CF65PU 155535300 IC50 = 0.03 nM T50594 C63TDJ 155535348 IC50 < 150 nM T50594 C29ORD 155535746 IC50 > 10000 nM T50594 CQ97VC 155535921 IC50 = 0.16 nM T50594 C3LC9I 155536820 IC50 = 792.3 nM T50594 C68GMW 155538446 IC50 = 43000 nM T50594 CX90PO 155538459 IC50 = 0.55 nM T50594 C6QY8K 155538969 IC50 = 0.02 nM T50594 C9J3IU 155538981 IC50 = 30 nM T50594 C68KHN 155539424 IC50 = 6.4 nM T50594 CXV14T 155539760 EC50 = 71 nM T50594 CI8JU5 155541036 IC50 < 150 nM T50594 C4H0LS 155541271 EC50 = 800 nM T50594 CWQ7F0 155541490 Ki = 1.3 nM T50594 CY8PB1 155542894 EC50 = 110 nM T50594 C2IG7U 155543022 IC50 = 3.1 nM T50594 CE03IU 155543981 IC50 = 92 nM T50594 CRG0K4 155544306 IC50 = 2.5 nM T50594 CPB87M 155545130 IC50 = 1.5 nM T50594 CNL4B8 155546196 IC50 = 4.5 nM T50594 CC83QJ 155547453 IC50 = 4.7 nM T50594 CEDN41 155550408 Ki = 0.4 nM T50594 CB73CQ 155551312 IC50 = 2.3 nM T50594 CG26ND 155552144 IC50 = 6.5 nM T50594 CORH39 155553574 EC50 = 220 nM T50594 CH18PL 155553803 EC50 = 215 nM T50594 CZQM57 155554194 IC50 = 511.8 nM T50594 CY6Q8S 155554337 IC50 = 18000 nM T50594 CG91LK 155555361 IC50 = 80 nM T50594 CXO5L1 155556907 EC50 = 2510 nM T50594 C6CJ3H 155557017 IC50 = 1.8 nM T50594 C62DJU 155558058 IC50 = 7.3 nM T50594 CU1MA5 155558576 EC50 = 915 nM T50594 CM0UH7 155559265 Ki = 1.2 nM T50594 C95EJG 155559459 IC50 = 0.35 nM T50594 CO2I4P 155559898 IC50 = 200 nM T50594 CG6T9Y 155559978 EC50 = 465 nM T50594 CRLP86 155560079 IC50 = 0.7 nM T50594 CJ9M3Y 155563039 IC50 = 0.9 nM T50594 C4EX3W 155563397 IC50 = 20.3 nM T50594 C46LPJ 155563540 EC50 = 330 nM T50594 CWN6O9 155565304 IC50 = 60 nM T50594 C43CBF 155566090 Ki = 0.9 nM T50594 C9WB2L 155566373 IC50 = 2.2 nM T50594 C1B7YH 155566566 IC50 = 0.7 nM T50594 CHCT58 155566705 IC50 > 10000 nM T50594 C04THL 155567360 Ki = 0.6 nM T50594 CUQ3O4 155567910 IC50 > 10000 nM T50594 CWE64A 155568407 IC50 = 7100 nM T50594 C4ED0G 155568443 IC50 = 1.5 nM T50594 CN38JC 155568642 IC50 = 433.71 nM T50594 CTZ24C 155568643 IC50 = 0.13 nM T50594 CV8W5R 155569485 Ki = 0.7 nM T50594 C13GYL 127031746 IC50 < 5000 nM T50594 D00ERW 44444843 Ki = 9182 nM T50594 D00HVA 11624601 Ki > 9200 nM T50594 D02XHC 448912 IC50 > 10000 nM T50594 D04ZTH 2817024 IC50 = 7520 nM T50594 D06HVH 54613583 IC50 = 60 nM T50594 D06UKS 44222958 IC50 = 1 nM T50594 D07MQC 9949093 IC50 = 1100 nM T50594 D07OXC 11650194 IC50 > 30000 nM T50594 D08HFG 24809764 IC50 > 10000 nM T50594 D09HVH 135566652 IC50 > 10 nM T50594 D09OWC 5373936 IC50 = 5100 nM T50594 D0F5EI 10017019 IC50 = 1000 nM T50594 D0L4WN 31420 IC50 = 24700 nM T50594 D0L6ND 10089677 IC50 = 10000 nM T50594 D0N3LC 90643548 IC50 > 1000 nM T50594 D0Q1HF 10521421 IC50 = 1280 nM T50594 D0Q3NG 11715520 Ki > 9200 nM T50594 D0RJ8J 76072859 IC50 > 1000 nM T50594 D0S7IE 11658882 Ki > 9200 nM T50594 D0T3PW 5281672 IC50 = 780 nM T50594 D0TO6S 2396 IC50 = 27 nM T50594 D0W7TU 947057 IC50 > 50000 nM T50594 D0X1RH 16051023 IC50 = 310 nM T25005 D03ZBT 11626560 IC50 > 10000 nM T25005 D04LVK 57379345 IC50 = 3360 nM T25005 D05NUH 54758501 IC50 = 1 nM T25005 D09KTS 24821094 IC50 = 0.1 nM T25005 D09PQZ 71226662 IC50 = 3.1 nM T25005 D0E6XR 3062316 IC50 = 1.3 nM T25005 D0OB0F 5328940 IC50 = 2.5 nM T25005 D0R3JB 4212 IC50 = 1000 nM T25005 D02TUL 118115473 IC50 = 607 nM T25005 D03LWG 53235510 IC50 > 10000 nM T25005 D04BFC 59174488 IC50 = 0.6 nM T25005 D07EHV 44814409 IC50 > 10000 nM T25005 D07HPJ 11476171 IC50 = 7600 nM T25005 D08AOZ 86582336 IC50 = 0.5 nM T25005 D0E3TC 44259 IC50 = 13.38 nM T25005 D0FD6D 11751922 IC50 = 93 nM T25005 D0G5XV 135565884 IC50 = 0.3 nM T25005 D0H0KH 54755438 IC50 = 5.2 nM T25005 D0O6WV 24794418 IC50 > 2000 nM T25005 D0QX8X 71479709 IC50 = 61 nM T25005 D0U7KH 86567195 Ki = 0.91 nM T25005 D0UT4W 135905454 IC50 = 0.63 nM T25005 D0YB3W 156414 IC50 = 185 nM T25005 D0Q1BE 72188716 IC50 = 6.5 nM T25005 D03FUO 25234918 IC50 = 14 nM T25005 D0T3ME 156422 IC50 > 30000 nM T25005 CR98MZ 613528 IC50 = 4100 nM T25005 C0ZI1F 2756534 IC50 = 15100 nM T25005 CI0P2J 2814562 IC50 = 3500 nM T25005 CXW3U6 3031415 IC50 > 6000 nM T25005 CPXK25 5793057 IC50 = 5150 nM T25005 CB7WK3 5938113 IC50 = 6700 nM T25005 CP0XI6 6603792 IC50 = 310 nM T25005 CM5Z8X 9869943 IC50 = 0.4 nM T25005 CSGD16 10246246 IC50 > 7000 nM T25005 C7SFI1 10296883 IC50 > 10000 nM T25005 CJ7U4I 11161778 IC50 = 23000 nM T25005 CW5C9X 11186250 IC50 = 1258.93 nM T25005 CRC86K 11397050 IC50 = 400 nM T25005 CM21YJ 11453049 IC50 = 1584.89 nM T25005 C7HMO6 11526786 IC50 > 10000 nM T25005 CACS26 11561968 Ki > 2000 nM T25005 CJ9KN7 11683817 IC50 > 10000 nM T25005 CU0E8O 11690457 Ki > 10000 nM T25005 C45EWD 11723489 IC50 > 7000 nM T25005 CP7AH3 11755812 IC50 = 7800 nM T25005 CS36BH 11843159 IC50 = 100 nM T25005 C2IS9W 11851477 IC50 = 150 nM T25005 CJXK96 11851580 IC50 = 60 nM T25005 CCN9L1 11851680 IC50 = 230 nM T25005 CJ6S2Q 11851879 IC50 = 30 nM T25005 C0FGK3 11852095 IC50 = 130 nM T25005 CF4S5D 11852469 IC50 = 21 nM T25005 CHR92S 11858109 IC50 = 27 nM T25005 C9RQN8 15950748 IC50 = 3423 nM T25005 C09OWB 16015442 IC50 = 1091 nM T25005 CKR57M 16086104 IC50 = 3330 nM T25005 C16NRY 16086114 IC50 = 545 nM T25005 CQG45C 16109001 IC50 = 25000 nM T25005 C5VPH9 16129448 IC50 = 4950 nM T25005 CL9BQ6 17748275 IC50 = 25000 nM T25005 CWH37T 17758574 IC50 > 10000 nM T25005 CAFW78 18450761 IC50 = 1954 nM T25005 C6BA1Y 18450866 IC50 = 767.5 nM T25005 CA61QF 21083895 IC50 = 17000 nM T25005 CFP37A 22347110 IC50 = 8.2 nM T25005 C6JV7W 23400934 IC50 > 7000 nM T25005 CD5S7O 23401001 IC50 > 7000 nM T25005 CK5N6B 23657635 IC50 = 97 nM T25005 CIZ4V1 24756997 IC50 = 9 nM T25005 C7YG1N 24759534 IC50 = 290 nM T25005 CQNP54 24764449 IC50 = 1000 nM T25005 C4Z9CN 24769780 IC50 = 126 nM T25005 CJUK39 24770517 IC50 > 10000 nM T25005 C9PA0M 24807809 IC50 > 10000 nM T25005 C9F1AO 24821023 IC50 = 0.5 nM T25005 CBW43O 24821811 IC50 = 20 nM T25005 CI5MQ1 24821812 IC50 = 0.58 nM T25005 CY48ZA 24821879 IC50 = 0.72 nM T25005 CY8L7E 24896769 IC50 > 10000 nM T25005 CIM4Q1 24901165 IC50 = 875 nM T25005 CFI7S2 24936376 IC50 = 13 nM T25005 C4KG6Z 24968331 IC50 = 42 nM T25005 CD5HQ0 24969301 IC50 > 10000 nM T25005 CD69RK 25097993 IC50 > 10000 nM T25005 C36FXD 25138012 IC50 = 9 nM T25005 CP6N4G 25138050 IC50 = 69 nM T25005 CSO82D 25154877 Ki = 0.25 nM T25005 CJL25F 25169253 IC50 = 5 nM T25005 C9Y0JV 25206375 IC50 = 8 nM T25005 CLH0V2 25234052 IC50 = 61 nM T25005 C1RU9T 25234054 IC50 = 1400 nM T25005 CKC10Q 25234136 IC50 = 88 nM T25005 C4D6UF 25234139 IC50 = 5 nM T25005 C2TPV7 25234524 IC50 = 6 nM T25005 C4MAC1 25234917 IC50 = 20 nM T25005 C6PQ7E 25234978 IC50 = 6 nM T25005 CNI4C8 25235043 IC50 = 3 nM T25005 C67VMP 25235106 IC50 = 20 nM T25005 C21DQU 25235170 IC50 = 5.9 nM T25005 CDU9Q6 25235171 IC50 = 9 nM T25005 CQD83X 25235172 IC50 = 14 nM T25005 C3L6ER 25235173 IC50 = 15 nM T25005 CZ64OU 25235174 IC50 = 9 nM T25005 CRO8T9 25263033 Ki = 125 nM T25005 CN5E0F 25263283 IC50 = 14000 nM T25005 CS2EW5 25264176 IC50 = 13 nM T25005 CK31XP 44182938 IC50 = 280 nM T25005 CB53SU 44182939 IC50 = 1600 nM T25005 CA98KR 44432441 IC50 > 22000 nM T25005 C6GP5Z 44548488 IC50 = 200 nM T25005 CLXZ05 44554064 IC50 = 38 nM T25005 C3VRO9 44557921 IC50 > 10000 nM T25005 C3XTA7 44562721 Ki = 78 nM T25005 C3HW7L 44570553 IC50 > 30000 nM T25005 C17PVE 44570554 IC50 > 30000 nM T25005 CLOY92 44570599 IC50 = 7000 nM T25005 CK06LT 44570600 IC50 > 30000 nM T25005 CMO3R5 44602494 IC50 = 30 nM T25005 C70VXL 44624435 IC50 = 144 nM T25005 CX0U3N 46220516 IC50 = 2 nM T25005 CB7WM8 46222818 IC50 = 10 nM T25005 C8JM5X 46223487 IC50 = 103 nM T25005 C0YTF8 46223725 IC50 = 132 nM T25005 CG71EF 46832441 IC50 = 327 nM T25005 C1LNX9 46832443 IC50 = 436 nM T25005 CH0JZ8 46833813 IC50 = 19 nM T25005 CD17VE 46833814 IC50 = 12 nM T25005 C9NCS8 46833815 IC50 = 11 nM T25005 C7H4YM 46865419 IC50 > 10000 nM T25005 CLS29B 46872626 IC50 > 10000 nM T25005 CZK6C2 46894111 IC50 = 8 nM T25005 CRB9E6 46908028 IC50 = 400 nM T25005 CF3Y7V 46908220 IC50 = 3 nM T25005 CKC0D5 46908221 IC50 = 2 nM T25005 CIG9W1 46908418 IC50 = 40 nM T25005 C9U6PT 46908706 IC50 = 50 nM T25005 CX9CT2 46909487 IC50 = 4 nM T25005 C9PAT7 46927672 IC50 = 10 nM T25005 C60GAV 46929544 IC50 > 8000 nM T25005 CP34VL 46929748 IC50 > 1000 nM T25005 CJ2E9Q 46929857 IC50 > 25000 nM T25005 CX65UM 49787738 IC50 = 2 nM T25005 C9L3XR 49838879 IC50 > 15000 nM T25005 CL4R0T 50925568 IC50 = 20 nM T25005 CI2VR3 51000608 IC50 = 4900 nM T25005 CDU90A 51000695 IC50 = 45000 nM T25005 C4P6MB 51000778 IC50 = 800 nM T25005 CWAX19 51000932 IC50 = 120 nM T25005 CR1W4B 51000933 IC50 = 1800 nM T25005 C5J4ZC 51000934 IC50 = 2300 nM T25005 CG8RL9 51000936 IC50 = 2700 nM T25005 CV0YT2 51000937 IC50 = 3200 nM T25005 CWOS84 51001012 IC50 > 10000 nM T25005 CO8UM9 51001094 IC50 = 200 nM T25005 CRNH80 51001177 IC50 = 100 nM T25005 C4E3LI 51001515 IC50 = 19000 nM T25005 C93AED 51001516 IC50 = 44000 nM T25005 CEQN27 52936621 Ki > 1000 nM T25005 C2W9OA 53324451 IC50 > 10000 nM T25005 C8ZRE3 53356518 IC50 = 8 nM T25005 C8NA4L 53384644 IC50 > 30000 nM T25005 CRD4Z6 54596323 IC50 = 8 nM T25005 CG1RK0 54596453 Ki = 0.69 nM T25005 CNH42M 54596723 Ki = 1.28 nM T25005 CM8JX1 56604907 IC50 = 10 nM T25005 CD3P6C 56644522 IC50 = 651.95 nM T25005 C6AN2Z 56656450 IC50 < 1 nM T25005 CJBL48 56925034 IC50 = 15 nM T25005 C18CKJ 56928445 IC50 = 3 nM T25005 C3KY5Z 56928861 IC50 = 3 nM T25005 CQGH97 57391046 IC50 = 13.2 nM T25005 C8GQ9H 57391143 IC50 = 1.55 nM T25005 CSU96R 57391144 IC50 = 76.5 nM T25005 C7OQ2B 57391145 IC50 = 13 nM T25005 C3X1ZN 57392910 IC50 = 3.33 nM T25005 COC5U3 57392911 IC50 = 1.89 nM T25005 CN03CZ 57392994 IC50 = 0.884 nM T25005 C2DRH3 57392995 IC50 = 19.1 nM T25005 CE1A9V 57394653 IC50 = 0.7 nM T25005 CIQH60 57394654 IC50 = 6.76 nM T25005 CD5Z9R 57394655 IC50 = 4.83 nM T25005 CNV76Z 57394656 IC50 = 2.6 nM T25005 CO34BP 57394657 IC50 = 40 nM T25005 C8W6IG 57395117 IC50 > 30000 nM T25005 CH2PZ8 57396405 IC50 = 6.58 nM T25005 CN8I2E 57396406 IC50 = 1220 nM T25005 C3NG0U 57396491 IC50 = 0.847 nM T25005 CNC84H 57396492 IC50 = 45.3 nM T25005 COG41M 57398104 IC50 = 7.56 nM T25005 C83EBV 57398105 IC50 = 60.6 nM T25005 CL78SU 57398205 IC50 = 12.2 nM T25005 CVRX72 57398206 IC50 = 9.53 nM T25005 C05PSA 57398207 IC50 = 72 nM T25005 CBK0C1 57399762 IC50 = 10.3 nM T25005 C4CQR0 57399857 IC50 = 5.51 nM T25005 COC32E 57401532 IC50 = 10.4 nM T25005 C7Z4PU 57401624 IC50 = 16.8 nM T25005 C7M2NU 57401629 IC50 = 1.82 nM T25005 CET8G9 57401630 IC50 = 5.35 nM T25005 C1CJ3Y 57401631 IC50 = 5.03 nM T25005 CCT87N 57401632 IC50 = 9.53 nM T25005 CDS7G4 57401633 IC50 = 670 nM T25005 C5THG9 57401721 IC50 = 2.52 nM T25005 C6LWX8 57401722 IC50 = 3.99 nM T25005 CU1C9S 57401723 IC50 = 4290 nM T25005 CZ4UR3 57403361 IC50 = 2.96 nM T25005 CY1Z7M 57403363 IC50 = 283 nM T25005 CG0Y3M 57403447 IC50 = 0.847 nM T25005 C3YGA0 57424138 IC50 = 3700 nM T25005 CG0O6Y 57473392 IC50 = 190 nM T25005 CNU76E 58043734 IC50 = 6 nM T25005 CD10RZ 58043863 IC50 = 81 nM T25005 C9JOQ3 58044026 IC50 = 4 nM T25005 C6J7QV 58044116 IC50 = 4 nM T25005 CY7N4D 58044297 IC50 = 1 nM T25005 CQEN24 58044306 IC50 = 2 nM T25005 CCF7Z0 58540029 IC50 = 4 nM T25005 C4KJL2 58540036 IC50 = 11 nM T25005 CPIF95 58540060 IC50 = 4 nM T25005 CMDI08 58540134 IC50 = 1 nM T25005 C68GRX 58540298 IC50 = 20 nM T25005 CR7WI1 58540323 IC50 = 4 nM T25005 CV13QY 58540422 IC50 = 3 nM T25005 CQ8VU9 58728932 IC50 = 8.9 nM T25005 C0EOY8 58729072 IC50 = 50 nM T25005 CCP4Z1 58729084 IC50 = 50 nM T25005 C94EVL 58729093 IC50 = 230 nM T25005 C1SI3L 59174579 IC50 < 1 nM T25005 COT79B 59216480 IC50 = 60 nM T25005 CT3EW2 59292007 IC50 > 1000 nM T25005 C2V9LI 59375017 IC50 = 9 nM T25005 C1L4FX 59375068 IC50 = 29 nM T25005 CBY4S3 59375142 IC50 = 11 nM T25005 CZ3TG1 59375154 IC50 = 16 nM T25005 CXJ63M 59603829 IC50 = 360 nM T25005 CQEU96 59603842 IC50 < 1 nM T25005 C1MR8Q 60097495 IC50 > 1000 nM T25005 CSZ6I5 66556035 IC50 = 251.19 nM T25005 C3ER5W 66601644 IC50 = 2 nM T25005 CD0LJ6 66604359 IC50 = 461 nM T25005 CT4RU2 66604890 IC50 = 189 nM T25005 C0JS8O 66604914 IC50 = 110 nM T25005 C0EVU7 66605043 IC50 = 379 nM T25005 CGS8J2 66605151 IC50 = 404 nM T25005 CCWU74 66605322 IC50 = 360 nM T25005 CN5BR8 66605844 IC50 = 308 nM T25005 CDES25 66606401 IC50 = 812 nM T25005 C9O2RZ 66895259 IC50 = 110 nM T25005 CSR94E 66895407 IC50 = 270 nM T25005 CQN0H3 66895621 IC50 = 70 nM T25005 CN7F2G 66926889 IC50 = 1 nM T25005 CW9RF7 67016212 Ki = 0.35 nM T25005 CKRX65 67016282 IC50 = 16700 nM T25005 CY9SL3 67016323 IC50 = 2600 nM T25005 C4U3XP 67016524 IC50 = 3 nM T25005 C1HSE0 67035086 IC50 = 580 nM T25005 CWI6K5 67035106 IC50 > 10000 nM T25005 C38RGB 67035556 IC50 > 10000 nM T25005 C37NKO 67129970 IC50 > 10000 nM T25005 CK80LJ 67130050 IC50 > 10000 nM T25005 CV63UL 67240318 IC50 > 10000 nM T25005 CR7DC4 67969461 IC50 < 100 nM T25005 CAF36T 67972044 IC50 = 9 nM T25005 C78QYC 67972152 IC50 < 100 nM T25005 C56FMK 67986337 IC50 < 100 nM T25005 CE4SM9 67986343 IC50 = 140 nM T25005 C7ARX2 67986346 IC50 = 460 nM T25005 CVZE42 67986349 IC50 = 550 nM T25005 C8C4ZF 67986352 IC50 = 400 nM T25005 CP7BO8 67986356 IC50 = 1200 nM T25005 CZY09U 67986357 IC50 = 1300 nM T25005 CZJ40Q 67986358 IC50 = 500 nM T25005 CLQ91B 67986410 IC50 > 10000 nM T25005 CLUR72 67986417 IC50 > 20000 nM T25005 CZNS75 68051325 IC50 < 100 nM T25005 C8I7GC 68293638 IC50 > 10000 nM T25005 CD56XK 68293660 IC50 > 10000 nM T25005 C7GRV2 68755406 IC50 > 10000 nM T25005 C5DGR9 69036886 IC50 = 1879 nM T25005 C3GTU1 69762142 IC50 > 10000 nM T25005 CY57QX 70647721 IC50 = 34 nM T25005 CD3A0B 70647727 IC50 = 3 nM T25005 C7VJ6A 70647728 IC50 = 2.6 nM T25005 C6E8DC 71092932 IC50 = 8600 nM T25005 CBKF84 71222614 IC50 = 0.3 nM T25005 C82IYH 71222927 IC50 = 10.7 nM T25005 CLIH32 71226367 IC50 = 0.3 nM T25005 CE4Y8J 71226521 IC50 = 11 nM T25005 CT4P8G 71226707 IC50 = 5.3 nM T25005 COU73Y 71226944 IC50 = 13 nM T25005 C15FZU 71227026 IC50 = 377 nM T25005 CSB2N6 71235464 IC50 = 3.3 nM T25005 C40JOZ 71235465 IC50 = 14 nM T25005 C5YX9S 71450146 IC50 = 2 nM T25005 CQR24F 71453784 IC50 = 1050 nM T25005 C6LH8Q 71455522 IC50 = 5 nM T25005 CL9YX8 71455523 IC50 = 12 nM T25005 C7C5KR 71459146 IC50 = 15 nM T25005 CO0U6L 71473856 IC50 = 8 nM T25005 CMEH30 71473900 IC50 = 5 nM T25005 CVET45 71473952 IC50 = 23 nM T25005 CPV31M 71473953 IC50 = 44 nM T25005 CH8NC9 71473954 IC50 = 9.9 nM T25005 C2PMJ7 71474167 IC50 = 4 nM T25005 C9U1ZP 71474168 IC50 = 0.8 nM T25005 CZ20PT 71474283 IC50 = 5.9 nM T25005 C8S2WR 71474333 IC50 = 290 nM T25005 CGL3O6 71474335 IC50 = 0.6 nM T25005 C6C0ED 71526523 Ki = 0.32 nM T25005 C9ILH0 71526524 Ki = 0.43 nM T25005 CC3JG4 71526687 Ki = 0.37 nM T25005 C1NPL0 71552941 IC50 > 30000 nM T25005 CA4PS8 71552942 IC50 > 30000 nM T25005 C3UA9C 71553011 IC50 = 30000 nM T25005 CEZ15Y 71553012 IC50 = 25670 nM T25005 CVIA91 71553085 IC50 = 30000 nM T25005 C1TR3O 71553152 IC50 = 30000 nM T25005 C8I9RX 71554042 Ki = 0.65 nM T25005 CAYK39 71555872 IC50 = 39 nM T25005 C7ZR4F 71555873 IC50 = 14 nM T25005 C82JZR 71555942 IC50 = 18 nM T25005 CK5L4A 71555944 IC50 = 8563 nM T25005 C05AUY 71555945 IC50 = 25 nM T25005 CA60YZ 71556002 IC50 = 20 nM T25005 CUOQ40 71556003 IC50 = 4946 nM T25005 CNVU70 71556004 IC50 = 166 nM T25005 CP0BZ1 71556006 IC50 = 11 nM T25005 CMAE80 71556057 IC50 = 47 nM T25005 CG7XR2 71556058 IC50 = 47 nM T25005 C3VRD2 71556060 IC50 = 24 nM T25005 CT1AB4 71556116 IC50 = 233 nM T25005 CC0W9V 71556633 IC50 = 16 nM T25005 CLO1K4 71556702 IC50 = 36 nM T25005 C79ITZ 71556766 IC50 = 208 nM T25005 C3S0AK 71556770 IC50 = 22 nM T25005 C3SCM1 71556835 IC50 = 48 nM T25005 C4TS8W 71557106 Ki = 1.3 nM T25005 C0DXC9 71558702 Ki = 6.3 nM T25005 C6C8KF 71558854 Ki = 1.8 nM T25005 C1UJA7 71558855 Ki = 6.9 nM T25005 CA0JH1 71559158 Ki = 0.43 nM T25005 C1SR5V 71576693 Ki = 3.2 nM T25005 C0I8ZY 71721544 IC50 = 0.67 nM T25005 C5O3GQ 71731698 IC50 = 6.4 nM T25005 CW0U1X 71731701 IC50 = 2.2 nM T25005 CS27TG 71731982 IC50 = 43 nM T25005 C4X1CP 71748056 Ki = 14.2 nM T25005 C1T5AI 71760912 IC50 = 1 nM T25005 CF04BD 71765399 IC50 = 850000 nM T25005 CZM1K4 71765510 IC50 = 5.6 nM T25005 C4KV0T 71765585 EC50 = 92 nM T25005 C5MJ0H 71765626 IC50 = 2 nM T25005 C6WU5A 71769203 IC50 = 5600 nM T25005 CKO8S6 71815907 IC50 = 13.5 nM T25005 CZU45Y 72165218 IC50 = 101 nM T25005 C5WYP9 72188715 IC50 = 8.3 nM T25005 C54XWG 72190869 IC50 = 3.1 nM T25005 CTA6P1 72191176 IC50 = 1.1 nM T25005 C46RQD 72191792 IC50 = 5.5 nM T25005 C0LAS6 72191795 IC50 = 1.2 nM T25005 C18RFO 72193307 IC50 = 6.8 nM T25005 CDWL69 72193608 IC50 = 21 nM T25005 C9TUP2 72201774 IC50 = 13 nM T25005 C9OQ2I 72710839 IC50 > 10000 nM T25005 CX75YR 73352604 IC50 = 316.23 nM T25005 CDNQ20 73388819 IC50 = 1.3 nM T25005 C0ZJV3 73389638 IC50 = 1.9 nM T25005 CVRQ65 73438218 IC50 = 6.6 nM T25005 CLQN18 73438269 IC50 = 1.08 nM T25005 CX87NM 73438270 IC50 = 3.76 nM T25005 CYML76 73438271 IC50 = 0.903 nM T25005 CE85VI 73438272 IC50 = 1.48 nM T25005 C2THR4 73438379 IC50 = 31.2 nM T25005 CF6QG1 73602845 IC50 = 7.15 nM T25005 CDN83F 73707530 Ki = 2 nM T25005 CX1LR9 73774633 IC50 = 0.25 nM T25005 CCQN01 73775788 IC50 = 25.3 nM T25005 CHF08G 73775789 IC50 = 79.1 nM T25005 COL37D 73775921 IC50 = 10.7 nM T25005 CVQW20 73775923 IC50 = 37.2 nM T25005 C5U4AF 73776059 IC50 = 16.3 nM T25005 CXW54V 73776061 IC50 = 16.4 nM T25005 CD83FL 73776204 IC50 = 38.6 nM T25005 CG84BR 73776205 IC50 = 17.4 nM T25005 C1P3DO 73776206 IC50 = 115 nM T25005 CN5D1R 73776207 IC50 = 6.01 nM T25005 CO1C8Y 73776208 IC50 = 12.3 nM T25005 CGC46K 73776360 IC50 = 24.5 nM T25005 CS9BQ1 74222426 IC50 = 21 nM T25005 CO0V6K 74222427 IC50 = 1.5 nM T25005 CBE71O 74222509 IC50 = 7.6 nM T25005 CM02PA 74222510 IC50 = 0.37 nM T25005 CWLT81 74222511 IC50 = 33 nM T25005 C4XSG8 74222512 IC50 = 0.41 nM T25005 CBT4M6 74222513 IC50 = 2.7 nM T25005 C53AFH 74222599 IC50 = 2.3 nM T25005 CDJ2U1 75203907 IC50 < 10 nM T25005 CBRK81 75204377 IC50 = 0.17 nM T25005 CF26RG 76901709 Ki = 1.2 nM T25005 CO3V8L 77844057 IC50 = 13 nM T25005 CY2I8Q 77844118 IC50 = 4.11 nM T25005 CRGK76 77844121 IC50 = 265 nM T25005 C4ISQ7 77844176 IC50 = 318 nM T25005 C1S9WZ 77844178 IC50 = 31 nM T25005 C0G9VL 77844179 IC50 = 222 nM T25005 C6DBN5 77844241 IC50 = 30.6 nM T25005 CN28TW 78318226 IC50 < 1 nM T25005 CCJ3P8 78318227 IC50 = 1.3 nM T25005 CQFR81 78318278 IC50 < 1 nM T25005 CBQ9L7 86276271 IC50 < 0.5 nM T25005 C3B1EZ 86280660 IC50 = 8 nM T25005 COD2E9 86294808 IC50 = 17000 nM T25005 C3OU4B 86302101 IC50 = 63 nM T25005 CPG3A5 86302574 IC50 > 30000 nM T25005 C1CBD9 86342498 IC50 = 20 nM T25005 C1M7NF 86342499 IC50 = 9 nM T25005 CE1VD9 86342500 IC50 = 28 nM T25005 CNZU96 86342680 IC50 = 37 nM T25005 CD2V1S 86342681 IC50 = 564 nM T25005 CT0BM6 86342682 IC50 = 124 nM T25005 CN43WE 86342683 IC50 = 472 nM T25005 C74DWF 86342866 IC50 = 254 nM T25005 CK1G0U 86567260 Ki = 1.8 nM T25005 CV0SZ5 86567261 Ki = 0.96 nM T25005 CI1QK2 86580532 IC50 = 1.2 nM T25005 CRA17V 86580533 IC50 = 0.27 nM T25005 CI30UB 86580691 IC50 = 1.5 nM T25005 CJ24PC 86580692 IC50 = 2.2 nM T25005 CN08AB 86580693 IC50 = 240 nM T25005 CZQR95 86582648 IC50 = 11 nM T25005 C50NMW 86582649 IC50 = 4 nM T25005 CR12AD 86699873 IC50 = 139 nM T25005 C3KJI6 86721755 IC50 = 9 nM T25005 CB7C6T 86721760 IC50 = 0.2 nM T25005 CJUZ46 86721780 IC50 = 160 nM T25005 CIJ5H0 86721782 IC50 > 100000 nM T25005 CPUW96 86721788 IC50 = 730 nM T25005 CW8I1N 86721789 IC50 = 18 nM T25005 CMK52I 86721807 IC50 = 2.1 nM T25005 C1IXU4 86721808 IC50 = 5.5 nM T25005 CN1KU6 86721813 IC50 = 1200 nM T25005 CZ5J3N 86721820 IC50 = 14 nM T25005 COA34E 86721822 IC50 = 9.9 nM T25005 CTYW83 86724331 IC50 < 10 nM T25005 CTY9E7 86762906 IC50 = 550 nM T25005 C02UGP 87056204 IC50 = 0.39 nM T25005 CR08QT 89266687 IC50 = 143 nM T25005 CV5XT9 89266735 IC50 = 1500 nM T25005 C98MTY 89266756 IC50 = 660 nM T25005 CHO8S0 89266780 IC50 = 1510 nM T25005 C39VWO 89266843 IC50 = 21 nM T25005 CN25CP 89285825 IC50 = 150 nM T25005 CSG38E 89455222 IC50 = 2.2 nM T25005 CT8I9U 89455387 IC50 = 23.9 nM T25005 C2LW7J 89548692 IC50 = 16.1 nM T25005 CW5YJ9 89548700 Ki = 0.8 nM T25005 C1HW4B 89735655 IC50 = 13000 nM T25005 C9MO1Y 89906279 IC50 < 10 nM T25005 C3YID4 89968957 IC50 = 3.2 nM T25005 CT18GX 89994856 IC50 = 1.9 nM T25005 CI5WT1 90001694 IC50 = 4 nM T25005 CTMO59 90008542 IC50 = 2.6 nM T25005 C3BL8D 90008602 IC50 = 6 nM T25005 C79KGU 90008606 IC50 = 5.1 nM T25005 C3T1UQ 90008615 IC50 = 11.7 nM T25005 CEF98J 90008863 IC50 = 5.4 nM T25005 C07CZK 90054287 IC50 = 1 nM T25005 CR3XL7 90119070 IC50 = 176 nM T25005 CLK3O0 90119255 IC50 = 170 nM T25005 CO2FV0 90119264 IC50 = 0.18 nM T25005 C3RL4C 90136268 IC50 = 61 nM T25005 C4ME0V 90136282 IC50 = 1.6 nM T25005 CY0T6O 90136348 IC50 = 3.7 nM T25005 CTPY64 90234618 IC50 = 101 nM T25005 CP4S1M 90244576 IC50 < 10 nM T25005 CJB9Q8 90283189 IC50 = 1.1 nM T25005 CD2VO4 90311700 IC50 = 294 nM T25005 CP0X1V 90311949 IC50 = 0.9 nM T25005 CJ27GT 90467690 IC50 = 2.3 nM T25005 CN7CG9 90644798 IC50 = 1106 nM T25005 CYAI75 90644799 IC50 = 2153 nM T25005 CLZ71J 90644800 IC50 = 133 nM T25005 C19HKY 90644801 IC50 = 304 nM T25005 C3MU1B 90644802 IC50 = 53 nM T25005 CI0VF7 90644803 IC50 = 52 nM T25005 COA7S0 90644804 IC50 = 8 nM T25005 CY5Z3V 90644805 IC50 = 15 nM T25005 CGIL57 90644806 IC50 = 14 nM T25005 CUDB61 90644807 IC50 = 1410 nM T25005 C4Q3ZA 90644808 IC50 = 45 nM T25005 CMZ01N 90644809 IC50 = 9 nM T25005 CXQ3V4 90644810 IC50 = 15 nM T25005 CA90YJ 90644811 IC50 = 15 nM T25005 CAH2N9 90644812 IC50 = 18 nM T25005 C7N6HP 90644813 IC50 = 11 nM T25005 CU03MC 90656042 IC50 = 67 nM T25005 CF0C1K 90656043 IC50 = 12700 nM T25005 CFQ97Y 90656044 IC50 = 150 nM T25005 C5M2LN 90656045 IC50 > 50000 nM T25005 CTAL51 90656046 IC50 > 50000 nM T25005 C5DV2G 90656047 IC50 = 38 nM T25005 CC5UO8 90656048 IC50 = 213 nM T25005 C1IA4Z 90656049 IC50 = 574 nM T25005 C3PJ2I 90656050 IC50 = 64 nM T25005 CQX17K 90656051 IC50 = 25 nM T25005 CY45AL 90656052 IC50 = 28 nM T25005 C39BDP 90656053 IC50 = 17 nM T25005 CDR9B1 90656054 IC50 = 143 nM T25005 CV6C8G 90656055 IC50 = 43 nM T25005 CX2P0H 90656056 IC50 = 87 nM T25005 CN1B9K 90656057 IC50 = 126 nM T25005 CZ5A9D 90656058 IC50 = 19 nM T25005 CL3MH1 90656059 IC50 = 170 nM T25005 CKO3R1 90656060 IC50 = 140 nM T25005 COI9D2 90656061 IC50 > 50000 nM T25005 CX3A5W 90656062 IC50 = 29000 nM T25005 CI9WR3 90656063 IC50 = 970 nM T25005 C2C6EQ 90656064 IC50 = 33 nM T25005 C8L4EH 90656065 IC50 = 65 nM T25005 C8UCD2 90656066 IC50 = 26 nM T25005 CP5E9X 90656067 IC50 = 32 nM T25005 CD4FM8 90656068 IC50 = 48 nM T25005 C9WO2A 90656069 IC50 = 83 nM T25005 CN9VX7 90656070 IC50 = 169 nM T25005 CZJB24 90656071 IC50 = 109 nM T25005 C9Y5CR 90656072 IC50 = 77 nM T25005 CPRI81 90656073 IC50 = 35 nM T25005 CM5F7W 90656074 IC50 = 18 nM T25005 C15HEM 90656075 IC50 = 49 nM T25005 CG9I7R 90656076 IC50 = 27 nM T25005 C4OB0T 90656077 IC50 = 41 nM T25005 CF89DA 90664659 IC50 = 15500 nM T25005 C90JVH 91799688 IC50 = 1.4 nM T25005 C6J0GR 91809511 EC50 = 28600 nM T25005 CED37U 91885524 IC50 = 15 nM T25005 C64SIO 92042864 IC50 = 794 nM T25005 C39PCS 101898032 IC50 = 4.8 nM T25005 CAKD54 102594000 IC50 = 75.6 nM T25005 C6TWN0 117668201 IC50 = 150 nM T25005 CM7C3W 117668218 IC50 = 17 nM T25005 CTK65N 117668270 IC50 = 8 nM T25005 C63LHQ 117668291 IC50 = 0.32 nM T25005 CP3VQ6 117668361 IC50 = 860 nM T25005 C0V3ZB 117676956 IC50 = 0.13 nM T25005 CO4Z3X 117676961 IC50 = 0.19 nM T25005 C7RUS2 117676973 IC50 = 0.15 nM T25005 CB4XM9 117676974 IC50 = 14 nM T25005 C3NI4J 117676976 IC50 = 0.36 nM T25005 C3AX9V 117676992 IC50 = 34 nM T25005 C5LWU4 117677006 IC50 = 0.8 nM T25005 CNOR97 117761007 IC50 = 2.6 nM T25005 CT8Y1R 117773317 IC50 = 1.1 nM T25005 CV69NM 117778362 IC50 < 0.3 nM T25005 C8Y5ZX 117778486 IC50 = 8.3 nM T25005 CIH2K3 117780573 IC50 = 2.5 nM T25005 C5B3CM 117781182 IC50 = 4.2 nM T25005 C30KSM 117781201 IC50 = 4.7 nM T25005 CT68XG 117785578 IC50 = 0.62 nM T25005 C7C6KO 117785630 IC50 = 4.3 nM T25005 C0EJ2H 117785631 IC50 = 4 nM T25005 CL91NV 117785647 IC50 = 1.6 nM T25005 C41YCU 117785685 IC50 = 3.8 nM T25005 C4K5WY 117785740 IC50 = 0.81 nM T25005 CSC8F7 117785816 IC50 = 34 nM T25005 CFZ0P3 117785848 IC50 = 15 nM T25005 CA0G4U 117787055 IC50 = 80 nM T25005 C2EKR6 117802839 IC50 = 2.1 nM T25005 C3FY8A 117838708 IC50 = 0.58 nM T25005 C7VDL3 117838709 IC50 = 0.53 nM T25005 C0BI1C 117838710 IC50 = 0.49 nM T25005 C73JCL 117838721 IC50 = 0.51 nM T25005 CT5L8Z 117925826 IC50 = 1.7 nM T25005 C8HYU9 117926195 IC50 = 2.6 nM T25005 C45OGJ 117926401 IC50 = 1.4 nM T25005 CPD57Q 117948653 IC50 = 0.4 nM T25005 CB4R8H 117948656 IC50 = 20.2 nM T25005 C34FKB 118025462 IC50 = 142 nM T25005 CUQS80 118025552 IC50 = 217 nM T25005 C1KGB4 118025559 IC50 = 584 nM T25005 CDF6L7 118025606 IC50 = 891 nM T25005 CGX1T6 118025676 IC50 = 7 nM T25005 C1IL8Q 118025680 IC50 = 86 nM T25005 C79ZBM 118025723 IC50 = 14 nM T25005 C6HO9P 118025760 IC50 = 67 nM T25005 CM4Z5V 118025790 IC50 = 1970 nM T25005 CX4W9A 118025823 IC50 = 104 nM T25005 C3FG4U 118025830 IC50 = 84 nM T25005 CM3JO2 118025835 IC50 = 123 nM T25005 CKR9G1 118025928 IC50 = 27 nM T25005 C5TQU3 118025943 IC50 = 12 nM T25005 C68YAU 118026010 IC50 = 43 nM T25005 CJ6ZB1 118038061 IC50 = 180 nM T25005 CQ0XS5 118038146 IC50 = 32 nM T25005 CZIS42 118038175 IC50 = 4.1 nM T25005 CZP8A2 118038240 IC50 = 0.09 nM T25005 CYC26N 118038298 IC50 = 4.4 nM T25005 C6O1JB 118038376 IC50 = 4.3 nM T25005 CFE6M2 118038416 IC50 = 0.8 nM T25005 C5HYV8 118038480 IC50 = 11 nM T25005 CC9W3M 118038535 IC50 = 25 nM T25005 C1RT3W 118038598 IC50 = 16.2 nM T25005 CXF0P7 118038619 IC50 = 1.9 nM T25005 CA3B9Z 118038785 IC50 = 500 nM T25005 CF8DV9 118039033 IC50 = 5900 nM T25005 C0D3QO 118039090 IC50 > 6000 nM T25005 CF31OY 118039156 IC50 = 430 nM T25005 C2WQ4G 118039220 IC50 = 2.3 nM T25005 CTU3K2 118043167 IC50 = 2.8 nM T25005 C32TIM 118043177 IC50 = 13 nM T25005 CMR1B0 118043198 IC50 = 1.3 nM T25005 CYQ54O 118043226 IC50 = 40 nM T25005 CPU7C0 118043263 IC50 = 1.9 nM T25005 CR2XJ5 118043265 IC50 = 1.3 nM T25005 CQ1L8G 118043278 IC50 = 10000 nM T25005 C4HQ5C 118043312 IC50 = 2.2 nM T25005 CB4A6H 118043313 IC50 = 1.6 nM T25005 CB40XP 118043323 IC50 = 0.5 nM T25005 CO0HE8 118107408 IC50 = 7.5 nM T25005 CE37KU 118107427 IC50 = 1.8 nM T25005 CJ1UV7 118107429 IC50 = 8.7 nM T25005 CTA7N8 118107436 IC50 = 0.9 nM T25005 C49LKY 118107459 IC50 = 5 nM T25005 C5VDB3 118107478 IC50 = 3.7 nM T25005 CR6ND3 118107479 IC50 = 32 nM T25005 CMX3U8 118107483 IC50 = 1.3 nM T25005 C0YW3E 118107484 IC50 = 86 nM T25005 CK9F4X 118107489 IC50 = 104 nM T25005 CYAD17 118107490 IC50 = 91 nM T25005 CJGT03 118346182 IC50 = 105 nM T25005 C02DGP 118346184 IC50 = 155 nM T25005 CU6NE2 118346192 IC50 = 19.1 nM T25005 CW25VP 118346194 IC50 = 17.7 nM T25005 CPJX70 118722806 IC50 = 1600 nM T25005 CPUT35 118722848 IC50 = 431 nM T25005 CA6KN9 118722849 IC50 = 1030 nM T25005 CT16GW 118722850 IC50 > 5000 nM T25005 CF59DR 118722851 IC50 = 818 nM T25005 CHD92M 118722852 IC50 = 171 nM T25005 COH06T 118722854 IC50 > 5000 nM T25005 C13XBH 118722855 IC50 > 5000 nM T25005 C48XIV 118727100 IC50 < 0.5 nM T25005 CM2HX1 118727101 IC50 = 0.5 nM T25005 C3F1AI 118728082 IC50 = 5.6 nM T25005 CVG7K0 118728083 IC50 = 3.2 nM T25005 C9V6TB 118728174 IC50 = 1568 nM T25005 C42HQG 118728175 IC50 = 79 nM T25005 COZ6D3 118728176 IC50 = 73.9 nM T25005 C8GAN5 118728177 IC50 = 58.3 nM T25005 CGR39I 118728178 IC50 = 135.5 nM T25005 C72MTN 118728179 IC50 = 41.7 nM T25005 CE39IR 118728180 IC50 = 15 nM T25005 CZUK91 118728340 IC50 = 4600 nM T25005 CF1I8Y 118728341 IC50 = 860 nM T25005 CXN4L5 118728342 IC50 = 225 nM T25005 CYIW78 118728343 IC50 = 40 nM T25005 CSDN72 118728344 IC50 = 30 nM T25005 CEZ9I1 118728345 IC50 = 90 nM T25005 CMF71L 118728346 IC50 = 150 nM T25005 CD1L2J 118728347 IC50 = 340 nM T25005 C7HNK8 118728348 IC50 = 190 nM T25005 CN4O3J 118728349 IC50 = 490 nM T25005 C25UBH 118728350 IC50 = 650 nM T25005 C6VLK2 118728351 IC50 = 43 nM T25005 CP8RC3 118728352 IC50 = 210 nM T25005 C3OIW8 118728353 IC50 = 54 nM T25005 CD3QC7 118728354 IC50 = 10 nM T25005 C2XI0G 118728355 IC50 = 60 nM T25005 CMY1F0 118728356 IC50 = 50 nM T25005 CO3EX8 118729088 IC50 = 4.3 nM T25005 CUX3Q5 118729089 IC50 = 7.8 nM T25005 C3HJC0 118729090 IC50 = 0.61 nM T25005 CGS36E 118729091 IC50 = 4.8 nM T25005 C13YHN 118729092 IC50 = 4700 nM T25005 CDKA65 118729174 IC50 = 10 nM T25005 C75QXY 118729175 IC50 = 50.8 nM T25005 C0JVF5 118729176 IC50 = 31.6 nM T25005 CR4WD5 118729177 IC50 = 12 nM T25005 CX0C5K 118729178 IC50 = 69 nM T25005 CTQ16U 118729179 IC50 = 118.8 nM T25005 CL7K5B 118729182 IC50 = 74 nM T25005 CR3A4I 118729183 IC50 = 1357 nM T25005 COR4G6 118729184 IC50 = 77.8 nM T25005 CWJ72S 118729185 IC50 = 46 nM T25005 C6D1WK 118729186 IC50 = 96.5 nM T25005 CGZ4S0 118729187 IC50 = 57.1 nM T25005 CS82YE 118729188 IC50 = 15.3 nM T25005 CF03VI 118729189 IC50 = 7 nM T25005 CYF9K8 118729190 IC50 = 25.2 nM T25005 CV42FJ 118729191 IC50 = 26 nM T25005 CFM07R 118729192 IC50 = 7.9 nM T25005 C47YUJ 118729193 IC50 = 11 nM T25005 COKJ09 118729194 IC50 = 69.7 nM T25005 CCWN20 118729195 IC50 = 574 nM T25005 C3X4GU 118729196 IC50 > 5000 nM T25005 CQCX41 118737057 IC50 = 67 nM T25005 CY8N5B 121293751 IC50 = 0.21 nM T25005 C12LTV 121293832 IC50 = 34 nM T25005 CX05DR 121293857 IC50 = 0.077 nM T25005 C37DUM 121293882 IC50 = 0.38 nM T25005 C86FHD 121293911 IC50 = 0.59 nM T25005 C9VM5J 121293927 IC50 = 81 nM T25005 C5VBP2 121293929 IC50 = 6 nM T25005 CU3Z6N 121293943 IC50 = 0.23 nM T25005 C1HKI5 121293949 IC50 = 0.11 nM T25005 CF7ZJ6 121293963 IC50 = 63 nM T25005 C0JQW1 121294046 IC50 = 1.2 nM T25005 CXQR89 121294143 IC50 = 0.14 nM T25005 CFS3E4 121294208 IC50 = 92 nM T25005 C4H3YT 121294217 IC50 = 12 nM T25005 C46DBJ 121362063 IC50 = 0.86 nM T25005 COGV39 121362167 IC50 = 0.39 nM T25005 CW4PG2 121362179 IC50 = 0.54 nM T25005 CO9SQ6 121454909 IC50 = 0.4 nM T25005 C63CXY 121454977 IC50 = 132 nM T25005 CH0X4Z 121454982 IC50 = 1 nM T25005 CD1S0Q 121455095 IC50 = 0.4 nM T25005 CNV26K 121455511 IC50 = 0.4 nM T25005 CYN8D9 121455521 IC50 = 0.1 nM T25005 CA59TF 121455523 IC50 = 0.2 nM T25005 C9ZTE0 121455568 IC50 = 1.3 nM T25005 C6XYK5 121455572 IC50 = 11 nM T25005 CBKR90 121455587 IC50 = 3 nM T25005 CT0KS4 121455652 IC50 = 0.2 nM T25005 CK78BX 121455673 IC50 = 26 nM T25005 C9OJ4T 121455700 IC50 = 0.3 nM T25005 C8XD1R 121455701 IC50 = 0.5 nM T25005 CW35TI 121455794 IC50 = 0.3 nM T25005 C6ZT2U 121455810 IC50 = 0.4 nM T25005 CT2JS5 121455892 IC50 = 0.2 nM T25005 C7CDN6 121468958 IC50 = 0.6 nM T25005 CG1SO6 121468959 IC50 = 0.4 nM T25005 C6YME4 121468960 IC50 = 3.4 nM T25005 C3XF0K 121468962 IC50 = 0.6 nM T25005 C1P9EV 121468963 IC50 = 0.2 nM T25005 C7OB1W 121468964 IC50 = 0.3 nM T25005 C0EFG1 121468967 IC50 = 2.5 nM T25005 CYO26S 121468970 IC50 = 0.6 nM T25005 CK03NG 121468972 IC50 = 309 nM T25005 CTFK25 121468974 IC50 = 13.9 nM T25005 CKZE17 121468976 IC50 = 62 nM T25005 CFM73S 121468978 IC50 = 0.8 nM T25005 CT2X7E 121481190 IC50 = 2.6 nM T25005 CZI09K 121499156 IC50 = 30 nM T25005 C7QE2J 121513893 IC50 = 421 nM T25005 CLPI09 122180346 EC50 > 50000 nM T25005 C6HKR2 122186249 IC50 > 10000 nM T25005 CL8UG5 122186250 IC50 > 10000 nM T25005 C0R5NS 122186251 IC50 > 10000 nM T25005 CC14AM 122186252 IC50 = 2295 nM T25005 CDUK97 122186253 IC50 > 10000 nM T25005 C6KWG4 122186254 IC50 > 10000 nM T25005 CHD5F2 122186255 IC50 = 1052 nM T25005 C9OWX5 122186256 IC50 = 107.4 nM T25005 CC41ON 122186257 IC50 = 176.2 nM T25005 C4P9NA 122186258 IC50 = 387.1 nM T25005 CD9E7X 122186259 IC50 = 699.2 nM T25005 CGQ1J9 122186260 IC50 = 279.7 nM T25005 C3J6BA 122186261 IC50 = 12.8 nM T25005 CKNF81 122186262 IC50 = 527.6 nM T25005 C7Y5EB 122186263 IC50 = 454.2 nM T25005 C7DW3G 122186264 IC50 = 291.5 nM T25005 C2SYA4 122186265 IC50 = 137 nM T25005 C84OGD 122186266 IC50 = 420.9 nM T25005 C4ZM7J 122186267 IC50 = 408.7 nM T25005 C8JT9S 122188509 IC50 = 12.2 nM T25005 CZN2V0 122188510 IC50 = 11.8 nM T25005 C7NJY1 122188511 IC50 = 9.5 nM T25005 C2LHC7 122188512 IC50 = 7.8 nM T25005 C5HY7G 122188513 IC50 = 7.4 nM T25005 CY5J4R 122188514 IC50 = 25.5 nM T25005 CLWJ56 122188515 IC50 = 54.9 nM T25005 CAJ19Q 122188516 IC50 = 21 nM T25005 CGRX10 122188517 IC50 = 9.9 nM T25005 C73RVY 122188518 IC50 = 1687 nM T25005 CH96TK 122188519 IC50 = 2867 nM T25005 CBS04E 122188520 IC50 = 3601 nM T25005 C0L9BY 122188628 IC50 = 455.7 nM T25005 C9P2HC 122188629 IC50 = 342.6 nM T25005 CNS5A6 122188630 IC50 > 10000 nM T25005 CJ27GC 122188631 IC50 = 2295 nM T25005 C1HUP9 122188632 IC50 = 1659 nM T25005 C8MBX1 122188633 IC50 = 853.9 nM T25005 C19LMB 122188634 IC50 = 183.3 nM T25005 CRB9U6 122188635 IC50 > 10000 nM T25005 C9M1ZH 122191198 IC50 = 16 nM T25005 CVWF79 122191199 IC50 = 28 nM T25005 CN0KS5 122191200 IC50 = 88 nM T25005 CD4RL5 122191223 IC50 = 39 nM T25005 CF2I6C 122191224 IC50 = 32 nM T25005 C4C9TS 122191225 IC50 = 30 nM T25005 C34CUW 122191226 IC50 = 55 nM T25005 CTC5D3 122191227 IC50 = 15 nM T25005 CDA73F 122191228 IC50 = 24 nM T25005 CS98FB 122191229 IC50 = 144 nM T25005 C02OZK 122191230 IC50 = 38 nM T25005 CU08AN 122191231 IC50 = 71 nM T25005 CO5T1L 122191232 IC50 = 59 nM T25005 C03BMP 122191233 IC50 = 103 nM T25005 CIS71B 122191234 IC50 = 44 nM T25005 CHR68P 122191235 IC50 = 127 nM T25005 C61RMU 122191236 IC50 = 101 nM T25005 C35WTN 122191237 IC50 = 13 nM T25005 CR5EC8 122191238 IC50 = 6.9 nM T25005 C1DN4E 122191239 IC50 = 32 nM T25005 C5J4PL 122191240 IC50 = 22 nM T25005 CFAY16 122191241 IC50 = 16 nM T25005 CLY87F 122191242 IC50 = 12 nM T25005 CN62UO 122191243 IC50 = 7.2 nM T25005 CH7P9T 122191634 IC50 = 3.8 nM T25005 CZY4G5 122191635 IC50 = 3.5 nM T25005 C6O2XI 122191636 IC50 = 9.4 nM T25005 CFKD32 122191637 IC50 = 3 nM T25005 CEY5J8 122191638 IC50 = 39 nM T25005 C4X7SD 122192466 IC50 > 10000 nM T25005 C0CGR8 122396707 IC50 = 6 nM T25005 C6JO4C 122474157 IC50 = 10.2 nM T25005 C0XB2E 122475292 IC50 = 15.1 nM T25005 C6QHB4 122484585 IC50 = 518 nM T25005 CRT93E 122484586 IC50 = 248 nM T25005 CF7ME6 122484587 IC50 = 982 nM T25005 CX8EC3 122484589 IC50 = 396 nM T25005 C2E8NC 122484594 IC50 = 145 nM T25005 CTX02B 122484677 IC50 = 996 nM T25005 CJ63LF 122484678 IC50 = 852 nM T25005 C6DP2N 122484680 IC50 = 6.2 nM T25005 C2SXK9 122484682 IC50 = 806 nM T25005 C8MJ4P 122484684 IC50 = 718 nM T25005 C1U2WJ 122484694 IC50 = 30 nM T25005 CJC73G 122484695 IC50 = 76 nM T25005 C4AUD3 122484700 IC50 = 359 nM T25005 CS58YZ 122484702 IC50 = 364 nM T25005 CX6KW7 122484733 IC50 = 349 nM T25005 CV63PN 122484734 IC50 = 0.8 nM T25005 C1NPL5 122484735 IC50 = 1.2 nM T25005 C01SPL 122484737 IC50 = 23 nM T25005 CME91S 122513214 IC50 = 0.7 nM T25005 C32TWI 122513222 IC50 = 12 nM T25005 CLM7K3 122604539 IC50 > 10000 nM T25005 C01JHI 122604566 IC50 > 10000 nM T25005 C6UY2L 122633880 IC50 > 10000 nM T25005 CC7P2W 122633900 IC50 = 437 nM T25005 C4E7VI 124176804 IC50 = 6.6 nM T25005 CGN3H7 127034237 IC50 = 5.65 nM T25005 CWQ5C6 127039627 IC50 = 6 nM T25005 CYXB27 127039628 IC50 = 6 nM T25005 CX8J3E 127043557 IC50 = 1070 nM T25005 C2OSC6 127044265 IC50 = 880 nM T25005 CW85CM 127044597 IC50 = 1320 nM T25005 C01ERK 127044779 IC50 = 70 nM T25005 C6H1GW 127045093 IC50 = 1800 nM T25005 CIU72D 127264586 IC50 = 24.5 nM T25005 CGQZ74 129048381 IC50 = 6873 nM T25005 C0XS4M 129896681 EC50 = 4.7 nM T25005 CGIT40 129896911 IC50 = 24 nM T25005 CFD38L 130247375 IC50 = 1000 nM T25005 CK8UP1 130247747 IC50 = 10 nM T25005 CJ01GR 130247785 IC50 <= 10 nM T25005 C9XE1Y 130247799 IC50 = 100 nM T25005 CART50 130248020 IC50 <= 10 nM T25005 CZYM59 130248042 IC50 <= 10 nM T25005 C3RP1U 130248888 IC50 >= 10000 nM T25005 C6NH7E 130271687 IC50 = 100 nM T25005 CXV7B5 130319034 IC50 = 89 nM T25005 C5LOI7 130362292 IC50 = 0.16 nM T25005 CB8X2L 130362298 IC50 = 59 nM T25005 CA46DB 130362493 IC50 = 0.46 nM T25005 C71KMN 130429150 IC50 = 1213 nM T25005 CSG8J3 130429224 IC50 = 334 nM T25005 C5PT1M 130429242 IC50 = 1380 nM T25005 C0UNO3 130429244 IC50 = 153 nM T25005 CGFK71 130429248 IC50 = 1.91 nM T25005 CEX8D1 130429250 IC50 = 526 nM T25005 C9J6ZK 130429255 IC50 = 271 nM T25005 C6OMB1 132204257 IC50 = 95 nM T25005 C36ZNH 132231744 IC50 = 1.1 nM T25005 C92EAB 132231777 IC50 = 0.079 nM T25005 C2WL6U 132231784 IC50 = 0.17 nM T25005 C87MJN 132231796 IC50 = 0.24 nM T25005 CT0ZP1 132231829 IC50 = 1.2 nM T25005 CQXU93 132231841 IC50 = 0.18 nM T25005 CV89JM 132231876 IC50 = 0.21 nM T25005 CU9P7O 132247592 IC50 = 4.5 nM T25005 CD6TW5 132550270 IC50 = 0.82 nM T25005 CRV07S 132597737 IC50 = 47.4 nM T25005 CGV9B8 134135637 IC50 = 112 nM T25005 C56UDO 134135820 IC50 > 100 nM T25005 CU7E8V 134136144 IC50 = 32.1 nM T25005 C9GWC2 134136895 IC50 = 10.6 nM T25005 CQ2B0H 134137093 IC50 = 11 nM T25005 C25WAP 134137307 IC50 = 0.4 nM T25005 CQ61HU 134137344 IC50 > 100 nM T25005 CX1DP2 134138676 IC50 = 1.23 nM T25005 CN1I6V 134140323 IC50 = 17.1 nM T25005 C0PN3R 134140590 IC50 = 19 nM T25005 CE43OI 134144225 IC50 = 0.5 nM T25005 C20RHY 134145268 IC50 = 2.6 nM T25005 C3KZV6 134146771 IC50 > 100 nM T25005 C0F7OT 134149340 IC50 = 410 nM T25005 C10LWI 134151050 IC50 > 100 nM T25005 C43FPY 134151089 IC50 = 0.5 nM T25005 C1C7PJ 134152686 IC50 = 63 nM T25005 CG8OY3 134153160 IC50 > 100 nM T25005 C5HMI8 134153342 IC50 = 21.6 nM T25005 CUD7A8 134155908 IC50 = 97.1 nM T25005 C8CXZ9 134156759 IC50 = 13.2 nM T25005 C59HOQ 134277578 IC50 = 4.4 nM T25005 C0PZ5R 134277599 IC50 = 2.59 nM T25005 C7PWJ2 134277617 IC50 = 0.33 nM T25005 CRA2H1 134277633 IC50 = 1.34 nM T25005 CXJ8I0 134277643 IC50 = 0.64 nM T25005 C02RIA 134277647 IC50 = 0.63 nM T25005 CGH42R 134277652 IC50 = 0.62 nM T25005 COA14U 134277654 IC50 = 0.46 nM T25005 CQK0B5 134277685 IC50 = 1.8 nM T25005 C6S8VC 134277696 IC50 = 0.53 nM T25005 C49PIO 134277748 IC50 = 0.95 nM T25005 CD7VK4 134277767 IC50 = 0.7 nM T25005 CZ5E6L 134277773 IC50 = 0.66 nM T25005 C2CFK7 134277780 IC50 = 2.11 nM T25005 C6E7LW 134277790 IC50 = 0.94 nM T25005 C6T7NW 134277796 IC50 = 0.41 nM T25005 CU8ZP5 134277800 IC50 = 1.09 nM T25005 CTR4K6 134277828 IC50 = 0.68 nM T25005 C3AVH9 134551003 IC50 = 3 nM T25005 C4H5TL 134551018 IC50 = 6.1 nM T25005 C4TVJ1 134551049 IC50 = 3.3 nM T25005 C6HZF3 134551056 IC50 = 5.3 nM T25005 CX2VZ9 134551058 IC50 = 2.8 nM T25005 CN75GU 134611727 EC50 = 13300 nM T25005 C54FXD 134957362 IC50 > 10000 nM T25005 CTJ48K 135524085 IC50 > 10000 nM T25005 CUT1W7 135524168 IC50 > 10000 nM T25005 CY4D8I 135566504 Ki = 636.5 nM T25005 CZFA70 135611366 IC50 = 456 nM T25005 CG3UZ1 135927974 Ki > 1000 nM T25005 CRK8E5 136391507 IC50 = 1.9 nM T25005 CF3W4I 136928070 IC50 = 1000 nM T25005 CR69AU 136928128 IC50 = 2.7 nM T25005 C03VDE 136928142 IC50 = 2 nM T25005 C2RB4H 136961397 IC50 = 38.8 nM T25005 CMS37R 136961398 IC50 = 21.3 nM T25005 CTAS87 136983688 IC50 = 0.58 nM T25005 C8M2DL 136983691 IC50 = 9.5 nM T25005 CMOH82 136983718 IC50 = 0.64 nM T25005 C1JSX0 136983721 IC50 = 4.2 nM T25005 CRE05Z 136983730 IC50 = 232.6 nM T25005 CMP62O 136983732 IC50 = 1.6 nM T25005 CB26DO 136983736 IC50 = 4.2 nM T25005 C9J5KZ 136983740 IC50 = 1.6 nM T25005 CN7W2C 136983741 IC50 = 1.9 nM T25005 CPM64E 136983746 IC50 = 1.3 nM T25005 CM2IO7 136983748 IC50 = 0.38 nM T25005 C0F7EY 136983756 IC50 = 41 nM T25005 CID2U4 136983757 IC50 = 200 nM T25005 C60HNV 136983761 IC50 = 3.5 nM T25005 C4EKW0 136983767 IC50 = 0.24 nM T25005 CY89MV 137071299 IC50 = 11 nM T25005 C5MZV6 137189918 IC50 = 10910 nM T25005 CMCD09 137189935 IC50 = 46510 nM T25005 CT8EV4 137226337 IC50 = 3180 nM T25005 CXC69T 137321158 IC50 = 862 nM T25005 C3Z4AT 137321159 IC50 > 10000 nM T25005 C81LGX 137349435 IC50 = 7.5 nM T25005 C0A9SP 137353877 IC50 > 10000 nM T25005 C8WQ3V 137354009 IC50 = 365 nM T25005 CX4UT6 137475232 IC50 = 86 nM T25005 CBN69K 137475234 IC50 = 667 nM T25005 CFXK71 137475248 IC50 = 1697 nM T25005 CS5L0F 137475249 IC50 = 34 nM T25005 CM6P8G 137475250 IC50 = 19 nM T25005 CXKD71 137475453 IC50 = 63 nM T25005 CNI4D8 137475454 EC50 > 100 nM T25005 C21HSQ 137475456 IC50 = 273 nM T25005 C6P5AL 137475459 IC50 = 282 nM T25005 C1KSZ6 137475463 IC50 = 5.8 nM T25005 CTA26W 137475470 IC50 = 41 nM T25005 CPY52K 137475474 IC50 = 21 nM T25005 CUG84N 137475477 IC50 = 2610 nM T25005 C2FT1L 137475480 Ki = 6 nM T25005 C4K2UA 137475509 IC50 = 57 nM T25005 CL87BX 137475510 IC50 = 1261 nM T25005 CB2TR5 137475511 IC50 = 32 nM T25005 C36CKU 137475515 IC50 = 596 nM T25005 CIR4W0 137475517 IC50 = 65 nM T25005 C8PJ7Z 137475518 IC50 = 197 nM T25005 CE1O2J 137475520 IC50 = 3187 nM T25005 CE4ZT1 137475623 IC50 = 3736 nM T25005 CKIX38 137475632 IC50 = 4996 nM T25005 CLB03V 137475634 IC50 = 210 nM T25005 C4RZ6J 137475648 IC50 = 114 nM T25005 C4RH2N 137475657 IC50 = 1426 nM T25005 CJ5D6T 137475692 IC50 = 127 nM T25005 CC8H2P 137475700 IC50 = 244 nM T25005 CW12VL 137475702 IC50 = 1191 nM T25005 C4GYH0 137475704 IC50 > 10000 nM T25005 CZP8B9 137475873 IC50 = 68 nM T25005 CRKA51 137475874 IC50 = 187 nM T25005 CZ6YO7 137475875 IC50 = 76 nM T25005 C6J7QN 137632048 IC50 = 2410 nM T25005 CH9WK1 137632228 EC50 = 1576 nM T25005 C6VN7C 137632252 IC50 > 100 nM T25005 C0S6PX 137632398 IC50 > 100 nM T25005 CM28ZT 137632791 IC50 = 1.18 nM T25005 C30SZG 137633174 IC50 = 6 nM T25005 CXT73R 137633588 IC50 = 132 nM T25005 CRLT63 137633687 IC50 = 4 nM T25005 CZOD53 137633880 IC50 = 0.25 nM T25005 CI1E8V 137634241 IC50 = 5020 nM T25005 C9QGJ0 137634325 IC50 > 10000 nM T25005 CCM5R7 137634499 Ki = 1.8 nM T25005 C86CNU 137634727 IC50 = 0.23 nM T25005 C3UGD5 137635118 IC50 = 68.3 nM T25005 C6LPM5 137635156 IC50 = 0.5 nM T25005 C5VQM1 137635526 IC50 = 231 nM T25005 CJKI16 137635532 Ki = 0.58 nM T25005 CR2K6M 137635680 IC50 = 9.14 nM T25005 CYM4L6 137635963 IC50 = 0.5 nM T25005 C7BJY5 137636807 IC50 = 0.59 nM T25005 C7IL4D 137637204 IC50 = 0.7 nM T25005 CU9YQ3 137637635 IC50 = 911 nM T25005 C39XGQ 137637902 IC50 = 38 nM T25005 CWZY04 137638548 Ki = 3.3 nM T25005 CH1Y2J 137639108 IC50 = 0.42 nM T25005 C3ABE0 137639720 IC50 = 0.2 nM T25005 C4VDL6 137640150 IC50 = 0.92 nM T25005 CJ28YI 137640151 IC50 = 350 nM T25005 C40XZN 137640550 IC50 = 21.3 nM T25005 CQOW35 137641160 IC50 > 100 nM T25005 C7FWD3 137641710 Ki = 0.45 nM T25005 CNL87M 137641918 IC50 = 85.4 nM T25005 CBJX42 137642666 IC50 = 5.9 nM T25005 CJVX98 137642896 IC50 = 18.1 nM T25005 C9XWS8 137643176 IC50 = 78.6 nM T25005 CEYA97 137643185 IC50 = 22.4 nM T25005 C4DRX1 137643187 IC50 = 5030 nM T25005 CW5V3F 137643326 IC50 = 1.4 nM T25005 C2ID4H 137643621 IC50 = 6.7 nM T25005 CF5DH3 137643910 IC50 > 5000 nM T25005 CQZ6N3 137644623 IC50 = 22.6 nM T25005 C4I8HP 137644728 Ki = 2.5 nM T25005 CFU7S2 137645034 Ki = 1.8 nM T25005 CVFR40 137645536 Ki = 1.8 nM T25005 C20MIC 137645538 IC50 = 7.12 nM T25005 C3GC8E 137646450 IC50 = 0.3 nM T25005 C3BP6L 137646652 IC50 = 110 nM T25005 CB6H7D 137646812 IC50 = 9.7 nM T25005 C4X7BG 137647868 IC50 = 0.3 nM T25005 CBYF68 137647965 IC50 = 9.5 nM T25005 CN8F6I 137648044 IC50 = 20 nM T25005 C96CMS 137648135 IC50 = 0.6 nM T25005 CO89DX 137649100 IC50 = 0.8 nM T25005 COLY80 137649218 IC50 = 0.1 nM T25005 C3FWY7 137649370 IC50 = 3.4 nM T25005 CAGB21 137649664 IC50 > 10000 nM T25005 C2QYK3 137649872 IC50 = 3 nM T25005 CYI4T1 137650386 IC50 = 2.83 nM T25005 C0D9MO 137651114 IC50 = 7.3 nM T25005 CH9W6N 137651389 Ki = 5.97 nM T25005 C7THC2 137652002 Ki = 4 nM T25005 CINE03 137652514 IC50 = 26 nM T25005 CBS5J3 137652658 IC50 = 27.2 nM T25005 C28QUP 137652864 IC50 = 88.6 nM T25005 C62JYT 137653234 IC50 = 91.3 nM T25005 C7R1WL 137653505 IC50 = 27.3 nM T25005 C6YAM7 137653900 IC50 = 69 nM T25005 C9T8NA 137654497 IC50 = 12.1 nM T25005 C1SWN5 137654673 IC50 = 1.05 nM T25005 C8BDX5 137655281 IC50 = 0.4 nM T25005 CU7I4L 137655908 IC50 = 48.6 nM T25005 COH9N2 137656066 Ki = 1 nM T25005 C6UW8I 137656158 IC50 = 5 nM T25005 C3YLU8 137656342 IC50 = 2946 nM T25005 CGW9I0 137656387 IC50 = 5000 nM T25005 C1T7DU 137656692 IC50 = 10.4 nM T25005 C3N4YM 137656842 IC50 = 213 nM T25005 CR6J9O 137656849 IC50 = 1.2 nM T25005 C7YHC0 137657046 IC50 = 58.5 nM T25005 CW1J7N 137657095 IC50 = 1.2 nM T25005 CF9Q8V 137657300 IC50 = 12.1 nM T25005 CV13JT 137657722 IC50 = 7.1 nM T25005 CJH0B6 137658413 Ki = 4.2 nM T25005 C03AHL 137658850 IC50 = 0.3 nM T25005 C0GC8I 137658926 IC50 > 10000 nM T25005 CRA21G 137658982 IC50 > 10000 nM T25005 CUP8I0 137659174 IC50 = 11 nM T25005 C2ZB5H 137660502 IC50 = 4.94 nM T25005 C40WUE 137660864 Ki = 1 nM T25005 C29HIS 137661280 IC50 = 28.3 nM T25005 CJ0SU5 137661571 IC50 = 23.8 nM T25005 CSTV07 137662233 IC50 = 92.7 nM T25005 CU2L5H 138108525 EC50 > 10000 nM T25005 CB8FE3 138393376 IC50 = 1 nM T25005 CN0X5D 138454787 IC50 = 161 nM T25005 CUXO19 138617501 IC50 > 1000 nM T25005 CRWA29 139030520 EC50 = 42.7 nM T25005 C72TXN 139465220 IC50 <= 10 nM T25005 CBI6F5 139465310 IC50 = 10 nM T25005 C47UIT 139473914 IC50 <= 10 nM T25005 C3JYA8 139474172 IC50 <= 10 nM T25005 C3JWI7 139507347 IC50 = 2.8 nM T25005 C1N5QZ 141366015 IC50 = 7 nM T25005 C9ZYG8 141366083 IC50 = 9.3 nM T25005 COW01B 141366090 IC50 = 2 nM T25005 CH5NU8 141366112 IC50 = 5 nM T25005 C5E3OG 141366257 IC50 = 16 nM T25005 C7RME6 141366266 IC50 = 3 nM T25005 C65RGZ 141366278 IC50 = 5 nM T25005 CIQ96U 141478757 IC50 = 1300 nM T25005 CLY5A8 141496674 IC50 = 209.2 nM T25005 C1OTX5 141496811 IC50 = 102.4 nM T25005 CZS03J 141509623 IC50 = 136 nM T25005 C32ADR 141509628 IC50 = 119 nM T25005 CHV69N 141509629 IC50 = 80 nM T25005 CS7F1P 141509631 IC50 = 183 nM T25005 CX12GN 141509638 IC50 = 106 nM T25005 CVG92Q 141509639 IC50 = 200 nM T25005 CV8MJ3 141509640 IC50 = 50 nM T25005 CU51PI 141531440 IC50 = 203.1 nM T25005 C81RPA 141531442 IC50 = 481.2 nM T25005 CAT46B 141531443 IC50 = 180.3 nM T25005 CSU0P6 141622000 IC50 = 5 nM T25005 CCX7L5 141622014 IC50 = 5 nM T25005 CF1R6Z 141725864 IC50 = 12.8 nM T25005 C6UA7H 142357225 IC50 = 2.1 nM T25005 CMHX97 145331319 IC50 = 1.9 nM T25005 CVID46 145331320 IC50 = 31.9 nM T25005 CW1P9K 145331325 IC50 = 17.2 nM T25005 CDB9Y1 145331327 IC50 = 5.4 nM T25005 CG6V5Q 145331334 IC50 = 20.8 nM T25005 CGPH07 145331338 IC50 = 236.6 nM T25005 C6C5DF 145331339 IC50 = 21.8 nM T25005 CXCO76 145331341 IC50 = 2.4 nM T25005 CFY21D 145961655 EC50 = 5790 nM T25005 CQ86LZ 145963345 EC50 > 10000 nM T25005 CJ38PD 145964020 IC50 = 417.4 nM T25005 CE9ML8 145964464 IC50 = 3.1 nM T25005 CPU95I 145964675 IC50 = 0.6 nM T25005 COXI60 145966049 IC50 = 8800 nM T25005 CO7Y6G 145966466 IC50 = 40 nM T25005 CZJ6K7 145966487 IC50 = 100 nM T25005 CA5T8S 145966795 IC50 = 52 nM T25005 CTJE41 145966905 IC50 = 6.1 nM T25005 C4OD9Q 145967187 IC50 = 0.4 nM T25005 C8C9KB 145967601 IC50 = 18.11 nM T25005 CAIB20 145967604 IC50 = 49.23 nM T25005 CS6G9N 145967737 IC50 = 15.9 nM T25005 CEK76M 145967834 IC50 = 11.3 nM T25005 CIR2O4 145968647 IC50 = 20.85 nM T25005 CI0XK9 145968683 IC50 = 0.5 nM T25005 CZT26F 145969236 IC50 = 10.95 nM T25005 C1U0NB 145969251 IC50 = 7.95 nM T25005 C4QH6O 145969743 IC50 = 26.89 nM T25005 CBDL98 145969762 IC50 = 18.1 nM T25005 CZ9I5X 145969766 IC50 = 9.84 nM T25005 CJR62Q 145970555 IC50 = 22.18 nM T25005 CF12YE 145970801 IC50 = 89.62 nM T25005 CN76WO 145970945 IC50 = 45.35 nM T25005 C0BGW8 145971022 IC50 = 725.2 nM T25005 C9T8HZ 145971801 IC50 = 0.4 nM T25005 C8NCR2 145971905 IC50 = 2.2 nM T25005 CB5HF9 145972552 IC50 = 23.8 nM T25005 C50WPS 145972838 IC50 = 40.1 nM T25005 CJB41K 145973790 IC50 = 7300 nM T25005 CA7X9N 145973949 IC50 = 22 nM T25005 CP2EY5 145974012 IC50 = 62.6 nM T25005 C8XAG3 145974040 IC50 = 3.7 nM T25005 CS6WP7 145974982 IC50 = 0.41 nM T25005 C1E0IL 145975398 IC50 = 440 nM T25005 C4M6OX 145976007 IC50 = 0.8 nM T25005 CM3D2W 145976100 IC50 > 1000 nM T25005 CU1OX3 145976315 IC50 = 23.6 nM T25005 C5WJ0D 145976790 IC50 = 4.3 nM T25005 CI8WD9 145977263 IC50 = 3.5 nM T25005 C3ISA8 145977288 IC50 = 4.3 nM T25005 C8S7YH 145977937 IC50 = 50.4 nM T25005 CIV26F 145978013 IC50 = 7.4 nM T25005 C4Z3BX 145978513 IC50 = 0.4 nM T25005 CXE8H0 145979687 IC50 = 17.1 nM T25005 CE31VG 145979714 IC50 > 10000 nM T25005 C5WH9O 145979909 IC50 = 0.52 nM T25005 CA2CD1 145980524 IC50 = 89.32 nM T25005 CR43KU 145980943 IC50 = 10.5 nM T25005 CNDI08 145981275 IC50 = 0.6 nM T25005 C4O7LK 145982512 IC50 = 0.82 nM T25005 CL3R7U 145982901 IC50 = 217 nM T25005 C34LTV 145982927 IC50 = 0.1 nM T25005 C5VF8P 145983087 IC50 = 126.4 nM T25005 C35FMR 145983116 IC50 = 8.7 nM T25005 C0YFS6 145983170 IC50 = 11.2 nM T25005 C48ZXP 145983545 IC50 = 8.7 nM T25005 C8O1AM 145983591 IC50 = 153 nM T25005 CA20KM 145983867 IC50 = 159 nM T25005 CN7W3R 145984041 IC50 = 9.1 nM T25005 CM8Z7V 145984082 IC50 = 6.5 nM T25005 CN4H3U 145984330 IC50 = 3.5 nM T25005 CVCP14 145984386 IC50 = 1.1 nM T25005 C52FGO 145984982 IC50 = 12 nM T25005 CG4U3I 145985120 IC50 = 420.4 nM T25005 C7EV2P 145985201 IC50 = 36 nM T25005 CXQ2O9 145985661 IC50 = 90 nM T25005 CT6P1E 145986054 IC50 = 2.4 nM T25005 CID7Y4 145986342 IC50 = 39.8 nM T25005 C3TH4Z 145986350 IC50 = 38.17 nM T25005 C17TBU 145986946 IC50 = 31.3 nM T25005 C52AOJ 145987765 IC50 = 1 nM T25005 CG9AH0 145987953 IC50 = 23.2 nM T25005 CM1K2H 145988251 IC50 = 8 nM T25005 C9BX4U 145988956 IC50 > 10000 nM T25005 CNI4C6 145989069 IC50 = 1600 nM T25005 CL1IV0 145989334 IC50 = 0.6 nM T25005 CGB2F6 145989547 IC50 = 0.7 nM T25005 C82FRH 145989705 IC50 = 0.8 nM T25005 CLM9U8 145989960 IC50 > 100 nM T25005 CQH40O 145990342 IC50 = 0.7 nM T25005 CMP97L 145990518 IC50 < 0.5 nM T25005 C6LSR8 145990895 IC50 = 0.8 nM T25005 C8T5QK 145991122 IC50 = 16 nM T25005 C8EAO1 145991760 IC50 = 1.6 nM T25005 C71HFI 145992300 IC50 = 81.7 nM T25005 CYZ72C 145994233 IC50 = 0.5 nM T25005 C3U4FY 155510736 IC50 = 5.68 nM T25005 C3EK1O 155510821 IC50 = 263.7 nM T25005 CMT02R 155511053 IC50 = 30.7 nM T25005 CS2U6K 155511219 IC50 = 18.5 nM T25005 CF27EG 155511610 IC50 = 287 nM T25005 CLAN63 155511649 IC50 = 23.7 nM T25005 CH3N4R 155512268 IC50 = 63.2 nM T25005 C3TAO2 155512304 IC50 = 2.39 nM T25005 C0AN1O 155512752 IC50 = 880 nM T25005 CB0N3M 155513186 IC50 = 56.9 nM T25005 C2MD1Q 155513187 IC50 > 10000 nM T25005 CA7O4B 155513491 IC50 = 8 nM T25005 C7MYO1 155514069 IC50 = 11.1 nM T25005 CZK4R0 155514194 IC50 = 35.6 nM T25005 CMR01Y 155514274 IC50 = 8.9 nM T25005 C7AMX8 155514903 IC50 = 942 nM T25005 CJ2XU8 155515191 IC50 = 11 nM T25005 C9PK2F 155515251 IC50 = 2229 nM T25005 CAR70X 155516363 IC50 = 36.6 nM T25005 CPM06N 155516429 IC50 = 35.4 nM T25005 CI23DH 155516489 IC50 = 996 nM T25005 C0GA2M 155516495 IC50 = 72.8 nM T25005 C5PHO9 155516709 IC50 = 154.5 nM T25005 CWXG94 155517099 IC50 = 8300 nM T25005 CLT70D 155517651 IC50 = 9.7 nM T25005 C8V9IM 155517893 IC50 = 68.3 nM T25005 CNBF94 155518187 IC50 = 7300 nM T25005 C4SVP7 155518257 IC50 = 38109 nM T25005 C6PT7H 155518445 IC50 = 13.2 nM T25005 C6Z8AT 155518957 IC50 = 130.6 nM T25005 C3NA2I 155519537 IC50 = 3 nM T25005 CL67JW 155520152 IC50 = 11.6 nM T25005 CGP0T7 155520658 IC50 = 16.5 nM T25005 C9TU2A 155520832 IC50 = 9.67 nM T25005 CI7HF6 155520873 IC50 > 500 nM T25005 C8HMN5 155521132 IC50 = 1.8 nM T25005 CC6O8T 155521339 IC50 = 2422 nM T25005 CD6BW4 155521972 IC50 = 258 nM T25005 C3MB7J 155522852 IC50 = 80.3 nM T25005 CLYQ13 155523828 IC50 = 125.2 nM T25005 CCF73Y 155524267 IC50 = 206 nM T25005 CFZ71B 155524499 IC50 = 15 nM T25005 CM09ZA 155524938 IC50 = 150 nM T25005 C9HBS1 155525156 IC50 = 45.5 nM T25005 C1TXJ8 155525159 IC50 = 159 nM T25005 C4O6HM 155525406 IC50 = 122.6 nM T25005 C1W5PI 155525516 IC50 = 6754 nM T25005 CRT67D 155526236 IC50 = 26 nM T25005 CE3OH1 155527121 IC50 = 35 nM T25005 CXOC93 155527452 IC50 = 18.4 nM T25005 CE2T0A 155527963 IC50 = 862 nM T25005 CIOL97 155528057 IC50 = 637 nM T25005 CZ1NG6 155528141 IC50 = 115.2 nM T25005 CG64WY 155528210 IC50 = 51 nM T25005 C5TY7L 155528304 IC50 = 2000 nM T25005 CCL2W7 155528484 IC50 = 1.15 nM T25005 CK5JY6 155528755 IC50 = 29.9 nM T25005 CTM92N 155528887 IC50 = 68000 nM T25005 CL38EX 155529541 IC50 = 2.3 nM T25005 CUXA18 155529935 IC50 = 1481 nM T25005 CM3Z8Q 155530172 IC50 = 3.6 nM T25005 CL0US4 155530459 IC50 = 3.9 nM T25005 C2WCU6 155530774 IC50 = 1456 nM T25005 C8WQY6 155531004 IC50 = 7.36 nM T25005 CQD8I0 155531565 IC50 = 8.49 nM T25005 CB1R7F 155531721 IC50 = 0.2 nM T25005 CMV9N8 155533061 IC50 = 1290 nM T25005 C0JNV2 155533438 IC50 = 27.1 nM T25005 C1NGV5 155534208 IC50 = 270 nM T25005 CM0U3I 155534552 IC50 > 1000 nM T25005 C1K8RJ 155534556 IC50 = 2.5 nM T25005 CZ81CR 155534707 IC50 = 8529 nM T25005 CS4A8R 155535551 IC50 = 213 nM T25005 C5TYF1 155535789 IC50 > 500 nM T25005 C78MZC 155536330 IC50 = 2 nM T25005 CD0R7C 155536414 IC50 = 98.2 nM T25005 CJ1IR4 155536431 IC50 = 8.21 nM T25005 C3LC9I 155536820 IC50 = 1584.89 nM T25005 CAQB79 155537002 IC50 = 11000 nM T25005 C2CG1A 155537016 IC50 > 10000 nM T25005 C06LXE 155538200 IC50 = 62845 nM T25005 CCN3M1 155538205 IC50 = 1.44 nM T25005 CNC60O 155538282 IC50 = 240.8 nM T25005 C3V4LG 155538413 IC50 = 237 nM T25005 C0U5YH 155538856 IC50 = 23 nM T25005 CBI81T 155539300 IC50 > 500 nM T25005 CW9J0A 155539317 IC50 = 14.8 nM T25005 CW6G3P 155540991 IC50 = 13.9 nM T25005 CFL16S 155541157 IC50 = 19000 nM T25005 CH10DU 155542091 IC50 = 1469 nM T25005 CZJ89B 155542162 IC50 = 4.2 nM T25005 CJXD07 155542870 IC50 = 10.8 nM T25005 C3FI9X 155543272 IC50 = 5254 nM T25005 CW73EO 155543439 IC50 = 36 nM T25005 C7K0OW 155544589 IC50 = 1120 nM T25005 CK6OS8 155545032 IC50 = 4195 nM T25005 C6F4JP 155546501 IC50 = 28.3 nM T25005 CDN60A 155547934 IC50 > 500 nM T25005 C1HPS7 155548524 IC50 = 21045 nM T25005 C4U9BD 155548652 IC50 = 73 nM T25005 CX9M1U 155548660 IC50 = 83.6 nM T25005 C4DC0V 155548954 IC50 = 733 nM T25005 C2Z4SX 155549111 IC50 = 23.3 nM T25005 C9Z7AM 155549842 IC50 = 91.7 nM T25005 CU94IA 155550455 IC50 = 125 nM T25005 C9VL3E 155550614 IC50 = 37114 nM T25005 CM9F6A 155551058 IC50 = 11.1 nM T25005 CFC2U1 155551386 IC50 = 90 nM T25005 CG7PR3 155552009 IC50 = 283.5 nM T25005 CE9UZ4 155552131 IC50 = 16000 nM T25005 CH0OY2 155552417 IC50 = 1.9 nM T25005 C6LEU2 155552459 IC50 = 4100 nM T25005 CHNU54 155552592 IC50 = 134 nM T25005 C0HUL3 155552710 IC50 = 434 nM T25005 C8TK4O 155552924 IC50 = 31.1 nM T25005 CPR9B5 155553418 IC50 = 2671 nM T25005 C8RFE7 155553522 IC50 = 18.8 nM T25005 CE0GX5 155554136 IC50 = 5169 nM T25005 C87XLB 155554564 IC50 = 105 nM T25005 CCK0F7 155554945 IC50 = 48.6 nM T25005 CX41VR 155556272 IC50 = 150 nM T25005 CM7Q3F 155556300 IC50 = 0.536 nM T25005 CHF87X 155557221 IC50 = 19155 nM T25005 C0FE4G 155557988 IC50 = 74 nM T25005 C21GNS 155558056 IC50 = 3.8 nM T25005 CHBD73 155558571 IC50 = 89.4 nM T25005 CZK10J 155558893 IC50 = 2096 nM T25005 CPAV79 155559005 IC50 > 3000 nM T25005 C9KX4D 155559215 IC50 = 550 nM T25005 C4L6HQ 155559509 IC50 > 10000 nM T25005 C51IBQ 155560019 IC50 = 1607 nM T25005 CY7FH8 155560115 IC50 = 614 nM T25005 C3HF6R 155561374 IC50 = 12000 nM T25005 CHT92X 155562269 IC50 = 7.8 nM T25005 C0OA5R 155562881 IC50 = 41.9 nM T25005 CW4LI7 155563694 IC50 = 27822 nM T25005 CW56DX 155563904 IC50 = 385.9 nM T25005 CAC85T 155564156 IC50 > 10000 nM T25005 C71ILK 155565394 IC50 = 617 nM T25005 C26URQ 155566212 IC50 = 45 nM T25005 CD0EK2 155566233 IC50 = 6.9 nM T25005 CPAY80 155566268 IC50 = 161 nM T25005 C9S8JX 155566610 IC50 = 333 nM T25005 CB8PM4 155567091 IC50 = 21888 nM T25005 C49EVT 155567502 IC50 > 500 nM T25005 CU0VN4 155567699 IC50 = 1437 nM T25005 CDW02C 155567865 IC50 = 8.58 nM T25005 CBE0S8 155568469 IC50 > 500 nM T25005 CGU74Q 155569301 IC50 = 286 nM T25005 C1ZE2Y 155569446 IC50 = 5323 nM T25005 CBP05X 155569566 IC50 = 0.9 nM T25005 D01RHR 71519693 IC50 = 5 nM T25005 D01VFR 4708 IC50 = 5830 nM T25005 D04PEI 11467730 IC50 = 4100 nM T25005 D06BJG 71556703 IC50 < 4.4 nM T25005 D07OXC 11650194 IC50 = 19 nM T25005 D0E7VO 59627005 IC50 = 3.5 nM T25005 D0GN5Z 5281295 IC50 = 6020 nM T25005 D0H3JH 24857323 IC50 = 0.61 nM T25005 D0N0LN 46908026 IC50 = 13 nM T25005 D0O6OH 71553154 IC50 = 950 nM T25005 D0OZ2S 11785878 IC50 = 410 nM T52522 D01UXC 2249 Ki = 9549.93 nM T52522 D02ZJI 123600 EC50 = 144.54 nM T52522 D03DJL 6918554 EC50 = 1.5 nM T52522 D03WEX 9966051 Ki = 560 nM T52522 D04JEE 4946 Ki = 0.32 nM T52522 D04KJO 3410 EC50 = 0.19 nM T52522 D04PHC 5816 Ki = 360 nM T52522 D04XEG 3343 Ki = 126 nM T52522 D05UVD 33624 Ki = 0.2089 nM T52522 D07MOX 439260 Ki = 3300 nM T52522 D0D1DI 3083544 EC50 = 0.3162 nM T52522 D0F2PO 4828 Ki = 0.4 nM T52522 D0G8NN 119570 Ki > 10000 nM T52522 D0I2MK 4171 Ki = 220 nM T52522 D0I8FI 3779 EC50 = 0.1585 nM T52522 D0K3ZR 2405 Ki = 250 nM T52522 D0K5CB 2083 EC50 = 25.12 nM T52522 D0L5YV 5152 EC50 = 0.07 nM T52522 D0M8RC 5403 EC50 = 3162.28 nM T52522 D0P1WA 5487427 EC50 > 10000 nM T52522 D0T7OW 681 Ki = 61000 nM T52522 D0X5NX 2783 Ki = 570 nM T52522 D0Y5AM 444031 EC50 = 0.7943 nM T52522 D0Z1WA 4916 Ki = 33 nM T52522 D04DJS 3682 Ki = 0.13 nM T52522 D06UKG 9849699 Ki = 0.012 nM T52522 D07WHS 5312115 Ki = 79200 nM T52522 D0A5EF 9887812 EC50 = 1258.93 nM T52522 D0DH5X 44472635 IC50 > 20000 nM T52522 D0G0RT 63952 EC50 = 0.76 nM T52522 D0GP8P 10372836 EC50 = 0.2512 nM T52522 D0H8OA 46917559 IC50 = 1700 nM T52522 D0I2XM 3038500 IC50 = 670 nM T52522 D0LI1C 44469321 IC50 > 10000 nM T52522 D0MT5C 16118894 IC50 = 120 nM T52522 D00OWF 5280953 Ki > 10000 nM T52522 D01SWK 5493324 EC50 = 13 nM T52522 D01VAB 2119 Ki = 0.5 nM T52522 D02KMG 9892481 EC50 = 0.0631 nM T52522 D04YJU 9829836 EC50 = 20 nM T52522 D05ZGW 5190 Ki = 57.3 nM T52522 D0AQ3H 11505444 EC50 = 0.26 nM T52522 D0C5PA 183812 EC50 = 0.631 nM T52522 D0G1RH 6918446 IC50 = 4.3 nM T52522 D0L5TJ 10527469 Ki = 3870 nM T52522 D0M7LV 5761 Ki = 740 nM T52522 D0Y1PG 9841972 EC50 = 290 nM T52522 D0ZG9N 132337 IC50 > 10000 nM T52522 C6TQ7E 2685 Ki = 1000 nM T52522 CYG2P9 2755 EC50 = 10000 nM T52522 CZUI83 2769 IC50 > 10000 nM T52522 CJQE97 5581 EC50 = 3.5 nM T52522 CS05VI 5807 EC50 = 128.82 nM T52522 C5H9CN 9287 Ki > 10000 nM T52522 C47EGS 56052 Ki = 180 nM T52522 CB6G3Z 91536 Ki = 0.54 nM T52522 CD3NO4 97803 Ki = 33800 nM T52522 CKP25M 121881 Ki < 1000 nM T52522 CZL87W 133999 IC50 > 10000 nM T52522 C96ASF 164451 Ki = 2350 nM T52522 C70UJK 183520 IC50 = 1600 nM T52522 C91DAE 185394 Ki = 0.88 nM T52522 CVUZ41 185395 Ki = 0.03 nM T52522 C8WG7P 203685 IC50 = 2.344 nM T52522 C0MOL1 204665 IC50 = 0.7244 nM T52522 CPA9F2 443372 EC50 = 6.31 nM T52522 C3LD8Q 688469 Ki = 3372.87 nM T52522 CF5QZ4 693141 Ki = 43200 nM T52522 CZN6S9 743974 EC50 > 31622.78 nM T52522 CVI84E 761003 Ki = 25118.86 nM T52522 CE6I2Y 913103 Ki = 9 nM T52522 CG53MQ 919019 Ki > 10000 nM T52522 CL8OU1 929854 Ki > 10000 nM T52522 C0LVU4 933006 Ki > 10000 nM T52522 CZF72W 1049240 Ki = 794328.23 nM T52522 CDZ6Q2 1070880 Ki = 39810.72 nM T52522 C2FKJ4 2299314 Ki = 9 nM T52522 CUM27P 2306318 Ki > 10000 nM T52522 C17WFV 2770390 Ki = 150 nM T52522 CRS35B 2796082 Ki = 700 nM T52522 CCY37O 2867500 Ki = 39810.72 nM T52522 CZ82ID 2967101 Ki = 1995.26 nM T52522 C4MXE1 2977358 Ki = 9 nM T52522 C7Z5OR 3086576 Ki = 320 nM T52522 CI32YO 3323563 Ki = 794.33 nM T52522 CZHG83 3416533 Ki > 100000 nM T52522 CD19NG 3654892 Ki = 110 nM T52522 CMSB89 3687256 Ki = 80 nM T52522 CT2A8D 3840250 Ki > 10000 nM T52522 CUEK98 3858663 Ki = 0.3 nM T52522 C9W6SB 3991311 Ki > 10000 nM T52522 CC9V5K 4013695 Ki > 100000 nM T52522 C1CK2S 4143663 Ki = 3290 nM T52522 CBC7N9 4276762 Ki = 300 nM T52522 CE1YN7 4292932 Ki = 23.5 nM T52522 CW2IR6 4421983 Ki = 80 nM T52522 C70GLP 5187268 Ki = 70 nM T52522 CCVA07 5484725 IC50 = 0.74 nM T52522 C23GIT 5767654 Ki = 9 nM T52522 CCX4I7 6460058 Ki = 9 nM T52522 CIZ7U3 6603820 Ki = 1200 nM T52522 CKP56W 6603867 Ki = 86000 nM T52522 C3A1FO 6604789 Ki < 10000 nM T52522 C1MW2P 6916441 EC50 = 13 nM T52522 CIQ70P 7334649 EC50 = 87.9 nM T52522 C7SIU5 9799092 EC50 = 50.12 nM T52522 CGX49B 9800339 EC50 = 1.4 nM T52522 CH6PX1 9801145 EC50 = 2511.89 nM T52522 CTN56U 9802994 IC50 = 300 nM T52522 CF1V5J 9803612 IC50 = 5011.87 nM T52522 C7ZQ3D 9803765 EC50 > 50000 nM T52522 C68VZH 9803988 EC50 > 10000 nM T52522 CRJ79X 9804536 EC50 = 353.1 nM T52522 C5FEX1 9804668 IC50 = 251.19 nM T52522 CT6JR1 9806791 Ki = 11.75 nM T52522 CUY3S0 9810596 IC50 = 7100 nM T52522 C7HQ9N 9816183 Ki = 5 nM T52522 CM48YW 9821129 Ki = 1600 nM T52522 CD7TA2 9823696 EC50 = 630.96 nM T52522 CD2U3O 9826638 IC50 = 540 nM T52522 CB6O2M 9827999 Ki = 74000 nM T52522 CYR8O6 9831168 EC50 = 36 nM T52522 CK7WI5 9832011 IC50 = 160 nM T52522 CK7DS2 9842600 EC50 > 10000 nM T52522 CS08ZV 9844005 IC50 = 280000 nM T52522 C3JYI0 9845280 EC50 = 501.19 nM T52522 C1CEO4 9845282 EC50 = 50.12 nM T52522 CHT1E3 9846763 IC50 = 1995.26 nM T52522 C0OS8W 9847067 EC50 = 0.5012 nM T52522 CY3DL8 9849126 EC50 = 0.1585 nM T52522 CTRI07 9852911 IC50 = 3000 nM T52522 C9FAP3 9853471 EC50 = 340 nM T52522 CB6R3T 9858463 Ki = 10 nM T52522 CZY34F 9860739 Ki = 3.75 nM T52522 CBD6E0 9866060 Ki = 382 nM T52522 CFVG52 9866061 Ki = 515 nM T52522 CN9YD5 9868131 IC50 = 4300 nM T52522 CJIR63 9871386 EC50 = 0.1259 nM T52522 CJ72CL 9871525 IC50 = 67 nM T52522 C1L6XP 9871887 Ki = 2.042 nM T52522 C51FVW 9872550 EC50 > 3160 nM T52522 CVF5O3 9873245 IC50 = 4 nM T52522 CSRF54 9873257 IC50 = 1600 nM T52522 CA43HC 9874175 EC50 = 0.36 nM T52522 CDQ84R 9888047 EC50 = 125.89 nM T52522 C5L3VF 9893058 EC50 = 1.259 nM T52522 CRV61G 9896742 EC50 = 37 nM T52522 CMC06V 9896817 EC50 = 1300 nM T52522 CYWQ50 9906447 Ki > 10000 nM T52522 C6CZ3G 9906777 IC50 > 10000 nM T52522 CQP6X3 9906822 EC50 = 5.2 nM T52522 CUHF02 9908924 Ki = 2250 nM T52522 C2A1CZ 9912443 EC50 > 1000 nM T52522 CMH72E 9912580 IC50 = 120 nM T52522 CDH69A 9915235 EC50 > 100000 nM T52522 CYH07G 9915238 IC50 = 3000 nM T52522 CGLY84 9917280 Ki = 1.514 nM T52522 CH9OT6 9917962 IC50 = 180 nM T52522 CW7YJ1 9924779 Ki = 30 nM T52522 C1XSL4 9927453 EC50 = 25 nM T52522 C10VOI 9930235 IC50 = 23 nM T52522 C4BVU7 9932018 EC50 = 0.3162 nM T52522 C92XMC 9933039 EC50 = 20 nM T52522 C7MO0Z 9938030 IC50 = 1660 nM T52522 CZM1E2 9946573 Ki = 37 nM T52522 C5VBO3 9956562 IC50 = 10000 nM T52522 CMI58L 9956563 IC50 = 14 nM T52522 CTL40E 9957764 EC50 = 0.02 nM T52522 CCN27K 9958539 EC50 = 1 nM T52522 CM6I4O 9960584 Ki = 66 nM T52522 CCA49K 9962058 IC50 = 100000 nM T52522 CB3AQ9 9967732 Ki = 21 nM T52522 CFTV18 9984028 EC50 < 1000 nM T52522 CIT57N 9985523 IC50 = 3000 nM T52522 CB8VU6 9986442 EC50 = 0.32 nM T52522 CZKM38 9992825 Ki = 580 nM T52522 C1NYC0 10002049 EC50 > 1000 nM T52522 C5KCI0 10006800 EC50 = 0.254 nM T52522 CO3DB4 10007337 IC50 = 3000 nM T52522 CP0H1B 10008017 EC50 = 80 nM T52522 C2S6LV 10027868 EC50 = 0.038 nM T52522 C2EUY0 10035109 Ki > 10000 nM T52522 CTE2I9 10048077 EC50 > 1000 nM T52522 CJP10L 10051943 Ki = 0.302 nM T52522 CWJ25B 10054165 IC50 = 760 nM T52522 CR73MA 10054373 EC50 = 14 nM T52522 CRU28L 10054896 IC50 = 7600 nM T52522 CBVG28 10075383 IC50 = 180 nM T52522 CVE2T1 10076176 EC50 = 1.995 nM T52522 C8TBK0 10076548 EC50 = 60 nM T52522 C7SL6M 10076885 IC50 = 2667 nM T52522 CAP5U7 10077662 EC50 = 0.687 nM T52522 CP7WF3 10092953 EC50 > 10000 nM T52522 CSNP15 10099346 IC50 = 1800 nM T52522 CL81PN 10099459 IC50 = 2300 nM T52522 CRK6B0 10101116 IC50 > 10000 nM T52522 CP6L3C 10112732 IC50 = 200 nM T52522 C8SAN2 10113837 EC50 > 100 nM T52522 CQW48U 10117815 Ki = 1500 nM T52522 CJ31XM 10119061 IC50 = 170 nM T52522 C07WRX 10121328 EC50 = 10 nM T52522 CKP0O1 10128077 EC50 = 0.5012 nM T52522 CCRO89 10132882 Ki = 120 nM T52522 CE27RV 10135864 EC50 > 10000 nM T52522 C8ZK3L 10138809 IC50 = 570 nM T52522 CZ0J7I 10140092 Ki = 510 nM T52522 CP0K9U 10140428 EC50 > 100000 nM T52522 C4B7XL 10140996 Ki = 1070 nM T52522 CO3F6S 10144004 EC50 > 100000 nM T52522 CCP74I 10160281 EC50 > 1000 nM T52522 C27MZY 10160636 IC50 = 400 nM T52522 CGJ10H 10162297 Ki = 350 nM T52522 C81STN 10173878 EC50 = 0.2512 nM T52522 CMK05F 10180590 EC50 = 0.1 nM T52522 C4YW9V 10202462 EC50 = 0.3162 nM T52522 C56USA 10203169 EC50 = 0.7943 nM T52522 C6Y5JB 10205362 IC50 = 140 nM T52522 CF5RL8 10206782 IC50 = 40 nM T52522 C2MX7I 10207208 Ki = 24 nM T52522 C1H0JA 10207209 Ki = 820 nM T52522 C3A2UK 10209243 EC50 > 10000 nM T52522 CF6R2U 10217757 EC50 = 0.1259 nM T52522 CPE8M6 10225563 EC50 = 0.3981 nM T52522 C2I6BY 10227108 Ki = 3100 nM T52522 C9Y4AT 10231679 Ki = 102 nM T52522 C2YDG7 10233153 EC50 = 60 nM T52522 CO64WJ 10236758 Ki = 43651.58 nM T52522 CSC3V2 10238776 EC50 = 0.7943 nM T52522 CDCP62 10239722 EC50 = 0.1 nM T52522 CW6C2I 10256921 EC50 = 0.258 nM T52522 CYBX59 10258518 IC50 = 1300 nM T52522 C1KR8D 10273469 Ki = 500 nM T52522 CV25SE 10278987 EC50 > 100000 nM T52522 C9TLW7 10282871 IC50 = 50 nM T52522 CO24KP 10283146 EC50 = 30 nM T52522 CF4Y7P 10283539 EC50 = 454 nM T52522 C9S2EY 10287658 EC50 = 3.981 nM T52522 C5TEI1 10288976 EC50 = 0.1585 nM T52522 C7F6LZ 10291064 Ki = 10 nM T52522 CD1S6J 10292413 Ki = 49 nM T52522 C2FSP4 10301101 EC50 > 100000 nM T52522 C3RP8X 10301445 EC50 > 1000 nM T52522 COES23 10304786 EC50 > 1000 nM T52522 CUML26 10305108 EC50 = 680 nM T52522 C42ZDS 10310047 EC50 = 1.259 nM T52522 COL3N7 10310564 EC50 = 1.995 nM T52522 CLO20K 10311070 EC50 = 1.259 nM T52522 C9Z1XJ 10324803 EC50 = 0.058 nM T52522 CG14VC 10326800 EC50 = 1.1 nM T52522 C0U7AV 10327461 EC50 = 0.5012 nM T52522 C9NQ0K 10327462 EC50 = 0.2512 nM T52522 C3E5CB 10337773 Ki < 100000 nM T52522 C1PSZ4 10346448 EC50 = 79.43 nM T52522 CZ26AE 10347866 IC50 = 12000 nM T52522 C0DTX5 10348864 EC50 = 2.6 nM T52522 C8QHR9 10349225 Ki = 8.71 nM T52522 C7H9PZ 10371216 IC50 = 980 nM T52522 CXI91M 10372344 EC50 = 0.2512 nM T52522 CGW4H2 10389119 EC50 = 0.051 nM T52522 C1QKW4 10390417 EC50 = 0.031 nM T52522 C3CLT1 10390752 EC50 = 0.058 nM T52522 CMR78G 10392857 EC50 = 0.122 nM T52522 CDRL02 10393774 EC50 = 5000 nM T52522 CR0V3S 10394806 EC50 = 0.1585 nM T52522 CA2N8B 10406968 Ki = 19 nM T52522 CF2ZN0 10411388 Ki = 9.2 nM T52522 CX0MO5 10414389 Ki = 1.549 nM T52522 C5QI3T 10416448 IC50 = 4700 nM T52522 C6URQ9 10416656 IC50 = 930 nM T52522 C38QCR 10431900 Ki = 220 nM T52522 C6ZIY2 10437614 IC50 = 110 nM T52522 C59OLP 10438390 IC50 = 1000 nM T52522 CA63EB 10438748 EC50 = 1.1 nM T52522 CA4PR8 10439505 EC50 = 0.5012 nM T52522 CBU5N3 10456417 Ki = 3.3 nM T52522 C6JY9O 10461973 EC50 = 0.1259 nM T52522 COV85C 10472143 Ki = 1100 nM T52522 CA20IB 10483845 IC50 = 21000 nM T52522 CRP7L9 10484263 EC50 = 8.4 nM T52522 CC3Z2P 10484922 EC50 = 0.5012 nM T52522 CQKI17 10544781 Ki = 616.6 nM T52522 C01LER 10548754 Ki = 6.457 nM T52522 CQ4Z8H 10553602 EC50 = 40 nM T52522 CL0MJ3 10553603 EC50 = 900 nM T52522 CK87QN 10575455 EC50 = 270 nM T52522 C9XUE2 10577317 Ki = 1.995 nM T52522 CB83SX 10601234 EC50 = 6000 nM T52522 C4NWL1 10602703 Ki = 3600 nM T52522 CW2S8I 10626150 EC50 = 3200 nM T52522 CWP9M1 10627736 IC50 = 980 nM T52522 C51DIX 10648298 EC50 = 4700 nM T52522 CX9WA0 10651078 IC50 = 760 nM T52522 C1C6KV 10651147 Ki = 480 nM T52522 CS4FX5 10697841 EC50 = 20 nM T52522 C8WX4M 10722793 IC50 = 1200 nM T52522 C6R5QN 10745501 EC50 = 10500 nM T52522 CFJA38 10746499 IC50 = 1800 nM T52522 C2MBK5 10789142 Ki = 7.762 nM T52522 C14SCL 10834286 Ki = 4365.16 nM T52522 CQA4E2 10841171 IC50 = 2600 nM T52522 CHM6J4 10841426 IC50 = 5000 nM T52522 C05CGB 10863093 EC50 = 19.95 nM T52522 C92OSW 10902809 EC50 = 10 nM T52522 CY1QM6 10940242 EC50 = 316.23 nM T52522 CNB39C 10947658 Ki = 4610 nM T52522 CC6V1Z 11002571 EC50 = 3162.28 nM T52522 CRJ5L3 11003341 EC50 = 398.11 nM T52522 C8V7XF 11005613 EC50 = 10 nM T52522 C6TAO1 11026016 EC50 = 5.012 nM T52522 CCKZ08 11038599 EC50 = 251.19 nM T52522 CZI9B1 11060184 EC50 = 31.62 nM T52522 C23NHX 11091850 EC50 = 1 nM T52522 C2N0BD 11124502 EC50 = 1000 nM T52522 C8FVK0 11134054 EC50 = 7.943 nM T52522 C34JRO 11169365 EC50 = 0.07943 nM T52522 CY04IB 11180293 EC50 = 0.1259 nM T52522 CQS49K 11188590 Ki = 76.6 nM T52522 COE80P 11189433 EC50 = 12.4 nM T52522 CRK79B 11214499 EC50 = 0.024 nM T52522 CB69KG 11224275 EC50 > 10000 nM T52522 CJ62RF 11247541 EC50 = 0.096 nM T52522 CM4AK7 11249243 EC50 = 0.027 nM T52522 CDM3U7 11259765 EC50 = 0.02 nM T52522 C3CY8X 11261001 EC50 = 0.04 nM T52522 CD2VF8 11268355 EC50 = 5.2 nM T52522 CBJ49T 11270071 EC50 = 330 nM T52522 CRFS12 11272641 EC50 > 10000 nM T52522 CC2Y4X 11299620 Ki = 40000 nM T52522 CJS9C0 11304851 IC50 > 25000 nM T52522 CJ4CE6 11324939 EC50 = 23 nM T52522 CQ08YH 11340895 EC50 > 10000 nM T52522 CGQ2D0 11342656 IC50 = 2000 nM T52522 CUNJ91 11352782 EC50 > 10000 nM T52522 CU9D3Q 11376125 EC50 = 0.056 nM T52522 C7Y3XZ 11398811 EC50 = 0.048 nM T52522 CM7E5J 11420492 EC50 = 0.064 nM T52522 CMX29E 11420551 EC50 > 10000 nM T52522 CQC36P 11432806 EC50 = 18 nM T52522 CL1M5W 11453340 EC50 > 1000 nM T52522 C4WMB3 11455274 EC50 = 0.023 nM T52522 CQS28E 11456127 EC50 = 0.066 nM T52522 C6TA1B 11476004 EC50 > 10000 nM T52522 CFC60E 11477877 EC50 = 0.032 nM T52522 CD2F7H 11489574 EC50 = 0.042 nM T52522 CBY69X 11489605 EC50 = 0.04 nM T52522 CW3YR2 11495581 EC50 = 1584.89 nM T52522 C16TWK 11508052 IC50 > 10000 nM T52522 CXWO08 11522273 IC50 > 10000 nM T52522 CF8L1D 11530695 IC50 = 1540000 nM T52522 C0Q8NC 11534330 EC50 = 0.17 nM T52522 CV6IN9 11539348 EC50 = 10.7 nM T52522 CZ62AI 11546349 EC50 = 1584.89 nM T52522 CAWR47 11556330 IC50 = 2300 nM T52522 CWGO05 11567751 EC50 = 3.4 nM T52522 CWM5K6 11575154 EC50 < 10000 nM T52522 CPG8V3 11577915 EC50 = 0.21 nM T52522 CP2WJ8 11592062 EC50 = 0.07943 nM T52522 CY15EM 11605652 EC50 = 10 nM T52522 C8A7SC 11617407 Ki = 0.4 nM T52522 C70VOJ 11621158 EC50 = 0.02 nM T52522 C12YSL 11625333 Ki = 175 nM T52522 C74VKM 11625493 EC50 = 15.4 nM T52522 CAU8C5 11625619 EC50 = 0.28 nM T52522 CKZ65X 11632691 EC50 = 58 nM T52522 CMIC92 11647002 EC50 = 0.25 nM T52522 C7ZTC8 11647543 EC50 = 1000 nM T52522 C1J4XV 11661536 EC50 = 3981.07 nM T52522 C1W6ZT 11668125 EC50 = 49.7 nM T52522 COHD32 11669967 EC50 < 10000 nM T52522 C24DOQ 11699773 EC50 = 0.045 nM T52522 CKJU26 11703823 EC50 = 1.3 nM T52522 CY9N5X 11707090 EC50 = 0.091 nM T52522 CZN5W9 11714238 EC50 = 0.24 nM T52522 CD31TA 11718543 EC50 = 10000 nM T52522 CPG15O 11743399 IC50 > 1000 nM T52522 CT1OL3 11758172 IC50 = 1700 nM T52522 C2UN8W 11785699 EC50 = 13 nM T52522 C4ISZ7 11810896 EC50 = 3.162 nM T52522 C85LXI 11857427 EC50 = 0.1995 nM T52522 C8JQL7 11957735 IC50 > 10000 nM T52522 C3BXJ2 12017001 IC50 = 3500 nM T52522 CF5TK1 12017002 IC50 = 21000 nM T52522 C38DZJ 12017003 IC50 = 3000 nM T52522 CN5A2D 12017004 IC50 = 4700 nM T52522 C40KFM 12017005 IC50 = 3700 nM T52522 C0G3XR 12017006 IC50 = 1400 nM T52522 C2FZ3H 12017007 IC50 = 2200 nM T52522 CDZQ57 12017010 IC50 = 3300 nM T52522 CEC98K 12017011 IC50 = 630 nM T52522 C02SVL 12017012 IC50 = 310 nM T52522 C1ZH0K 12017013 IC50 = 9000 nM T52522 C31JDV 12017014 IC50 = 940 nM T52522 CLIX97 12017015 IC50 = 2500 nM T52522 CO0ST4 12017016 IC50 = 320 nM T52522 C7Z8WC 12017017 IC50 = 3500 nM T52522 C60OVP 12017018 IC50 = 20000 nM T52522 CPU75A 12043155 IC50 = 1000 nM T52522 C1MFE0 12043156 IC50 = 962 nM T52522 CR0T9I 12043157 IC50 = 660 nM T52522 C4U9KY 12043158 IC50 = 44000 nM T52522 CW0XL2 12043159 IC50 = 57000 nM T52522 C7I2CM 12049914 IC50 = 8800 nM T52522 C5M8FQ 12049915 IC50 = 9300 nM T52522 C49XHR 12049916 IC50 = 1300 nM T52522 C7TAQ6 12049917 IC50 = 2500 nM T52522 CDI75Z 12049918 IC50 = 1600 nM T52522 C0LF7J 12049919 IC50 = 380 nM T52522 C6JWS8 12049920 IC50 = 780 nM T52522 CU7A5R 12049921 IC50 = 5000 nM T52522 CDZF95 12049922 IC50 = 860 nM T52522 CZ4V2K 12049923 IC50 = 8800 nM T52522 C8DUY7 12049924 IC50 = 690 nM T52522 CF0IG7 12049925 IC50 = 730 nM T52522 C3U1SP 12049926 IC50 = 620 nM T52522 CLD32O 12093446 EC50 = 0.3981 nM T52522 CNG9S3 12475776 Ki = 20400 nM T52522 CJBZ81 12972976 IC50 = 19952.62 nM T52522 CO8BW3 13208878 IC50 = 46.77 nM T52522 CZI4G6 13208884 IC50 = 74.13 nM T52522 C03EXV 13345218 EC50 = 0.1 nM T52522 CH0IF1 13699248 IC50 > 10000 nM T52522 CFC0D6 14823035 Ki = 3.2 nM T52522 CMO81H 14925759 Ki = 35481.34 nM T52522 C7JV1Z 15054187 Ki > 100000 nM T52522 C5RM1O 15054189 Ki = 1181 nM T52522 C7Z4YC 15054190 Ki > 100000 nM T52522 CKVQ30 15054191 Ki > 100000 nM T52522 CEBL08 15054192 Ki > 100000 nM T52522 CKFL78 15221053 Ki = 1230 nM T52522 C9HLK1 15221055 Ki = 11400 nM T52522 CLR24K 15461453 Ki = 5.4 nM T52522 C25CVZ 15483879 IC50 = 4000 nM T52522 CLNE19 15483880 IC50 = 2500 nM T52522 CUK85J 15483883 IC50 = 7500 nM T52522 CSDO83 15523859 IC50 = 380 nM T52522 C6Q9FZ 15523860 IC50 = 5000 nM T52522 CKP61A 15523861 IC50 = 2000 nM T52522 C1VWH5 15580747 Ki = 7700 nM T52522 C8U2XV 15981386 EC50 = 0.1995 nM T52522 CHW2T0 16035175 EC50 = 7.943 nM T52522 CKQ40B 16035281 EC50 = 7.943 nM T52522 C9MTH2 16035375 EC50 = 7.943 nM T52522 CKV03I 16035377 EC50 = 6.31 nM T52522 C8F7JQ 16035379 EC50 = 6.31 nM T52522 CB2M7O 16036676 EC50 = 10 nM T52522 CCTM64 16049024 EC50 = 0.1 nM T52522 C17ZSM 16049026 EC50 = 0.1259 nM T52522 CC3O5H 16049028 EC50 = 0.07943 nM T52522 C71EWF 16049029 EC50 = 0.1259 nM T52522 C3OC9G 16049087 EC50 = 0.0631 nM T52522 CD41WM 16049088 EC50 = 0.07943 nM T52522 C63MIJ 16049090 EC50 = 0.7943 nM T52522 C8B4VS 16049158 EC50 = 3.981 nM T52522 CE85LR 16049160 EC50 = 12.59 nM T52522 C27VPK 16049162 EC50 = 3.162 nM T52522 C6Z4CS 16049234 EC50 = 0.631 nM T52522 C7H8AV 16049289 EC50 = 0.7943 nM T52522 CP06JS 16049309 EC50 = 0.3981 nM T52522 CFC03X 16049361 EC50 = 3.981 nM T52522 CZ57RV 16049363 EC50 = 3.981 nM T52522 CB3MN6 16049374 EC50 = 1.259 nM T52522 C4QJE9 16049376 EC50 = 1.585 nM T52522 C19EUK 16049377 EC50 = 0.5012 nM T52522 CKY42H 16049448 EC50 = 1.585 nM T52522 CC4F0L 16049450 EC50 = 1 nM T52522 CH8KY4 16126657 EC50 > 10000 nM T52522 C42ELY 16219010 EC50 = 50.12 nM T52522 CERP08 16219807 Ki < 10000 nM T52522 C9JE3V 16222317 EC50 = 12.1 nM T52522 CDV38P 16222840 EC50 > 10000 nM T52522 C9ONT1 16222940 EC50 = 3200 nM T52522 CZ2IS9 16660294 Ki > 10000 nM T52522 C2P0SB 16717791 Ki = 261 nM T52522 CIC38O 16735257 EC50 = 0.3 nM T52522 C6Y9LU 16735259 EC50 = 33.2 nM T52522 C0UXI1 16735261 EC50 = 7.2 nM T52522 CR0VT9 16735263 Ki = 6025.6 nM T52522 C05FHR 16735272 EC50 = 2.7 nM T52522 CC0NY4 16735492 Ki = 28800 nM T52522 CKZI13 16735493 Ki = 30800 nM T52522 CM5D7A 16735494 Ki = 22908.68 nM T52522 C4FVP7 16735495 EC50 = 12.5 nM T52522 C01KQT 16736091 EC50 = 2 nM T52522 CO5U6P 16736092 Ki = 28600 nM T52522 CUE3O4 16736094 Ki = 1860 nM T52522 C5GTV9 16736096 Ki = 1778.28 nM T52522 C31SJZ 16736514 Ki = 20417.38 nM T52522 C9WFR6 16737369 Ki = 2511.89 nM T52522 CZ7BM5 16737411 Ki = 2930 nM T52522 C0C5RO 16737412 Ki = 7940 nM T52522 CWM76C 16737588 Ki = 10471.29 nM T52522 CHRG71 16738927 EC50 = 0.1995 nM T52522 CD3OE5 18525747 Ki = 33500 nM T52522 CK4TR0 19082200 EC50 = 0.5012 nM T52522 CWJ7K6 19360455 IC50 = 21 nM T52522 C9JD5Y 19360456 IC50 = 21 nM T52522 CMW4X0 21093243 IC50 = 19952.62 nM T52522 CTR6Z3 21435491 IC50 = 7943.28 nM T52522 C3T5HF 21509921 Ki > 10000 nM T52522 C1JBM4 22063464 EC50 = 4.1 nM T52522 CT34YN 22712045 EC50 = 0.3981 nM T52522 C0M9SR 22986860 IC50 = 251.19 nM T52522 CN9Z2S 23661589 EC50 = 794.33 nM T52522 CIP94M 24229559 IC50 = 10000 nM T52522 CWEM23 24321330 Ki = 230 nM T52522 C1V2UI 24764458 EC50 = 3.7 nM T52522 CHI83W 24769038 IC50 > 30 nM T52522 C7QK6D 24804878 EC50 = 0.4 nM T52522 CST3O6 24822310 EC50 > 1000 nM T52522 CVH1N4 24822974 EC50 > 1000 nM T52522 CBS82N 24823127 EC50 > 1000 nM T52522 CHDE90 24823464 EC50 = 586 nM T52522 C3HK0J 24865725 Ki = 501.19 nM T52522 C0O6FX 24865727 Ki = 1584.89 nM T52522 CI65LR 24876564 EC50 = 129 nM T52522 C43RTZ 24882193 IC50 > 10000 nM T52522 C8ABL2 24882564 IC50 = 15000 nM T52522 CR6N2C 24885648 Ki = 9 nM T52522 C1SFL2 24886595 Ki = 55 nM T52522 C08VXN 24893964 EC50 > 1000 nM T52522 CI53SE 24893978 Ki > 10000 nM T52522 CYN9K4 24894127 EC50 > 10000 nM T52522 C5AD3B 24895261 EC50 > 10000 nM T52522 CW8V3F 24895263 EC50 = 1100 nM T52522 CT7AM8 24895361 EC50 > 10000 nM T52522 CIOG69 24895783 EC50 > 1000 nM T52522 CLV98U 24895789 EC50 > 1000 nM T52522 CA08KY 24900423 EC50 = 10 nM T52522 CG15KX 24900424 EC50 = 0.631 nM T52522 C13JLE 24900426 EC50 = 0.5012 nM T52522 C1U9VL 24900685 EC50 = 0.5012 nM T52522 CU3F7K 24900689 EC50 = 0.631 nM T52522 CPLO51 24900749 EC50 = 3.162 nM T52522 CX69CF 24900750 EC50 = 0.7943 nM T52522 CE5W9U 24900751 EC50 = 3.162 nM T52522 CQDR84 24900811 EC50 = 3.162 nM T52522 CIL8Q7 24900812 EC50 = 0.631 nM T52522 C9YUP8 24900813 EC50 = 0.631 nM T52522 C63ILV 24900872 EC50 = 1 nM T52522 CSF3J2 24900874 EC50 = 15.85 nM T52522 C4AT0P 24900937 EC50 = 0.631 nM T52522 C2NR7M 24900942 EC50 = 0.3981 nM T52522 C58DZC 24901140 EC50 = 1 nM T52522 CW0QV2 24901141 EC50 = 0.5012 nM T52522 CHWE43 24901143 EC50 = 0.3162 nM T52522 C5ZCX4 24901144 EC50 = 0.1585 nM T52522 CNP40V 24901209 EC50 = 0.3162 nM T52522 C7MGC9 24901210 EC50 = 0.2512 nM T52522 CS6BH7 24901211 EC50 = 0.3162 nM T52522 C4JB7G 24901283 EC50 = 1.995 nM T52522 CBS0V5 24901284 EC50 = 1.259 nM T52522 C83MAF 24901285 EC50 = 0.7943 nM T52522 CVE24O 24901347 EC50 = 0.2512 nM T52522 CV5GY0 24901348 EC50 = 0.3162 nM T52522 CFZ5D7 24901349 EC50 = 0.3981 nM T52522 CCMQ16 24901351 EC50 = 0.3162 nM T52522 CGW2U6 24901413 EC50 = 0.2512 nM T52522 COY5H0 24901416 EC50 = 1.585 nM T52522 C4BU6R 24936488 Ki = 2600 nM T52522 CH87SX 24936489 Ki = 81 nM T52522 CIR69S 24936491 Ki = 175 nM T52522 C75UCO 24936492 Ki = 28 nM T52522 CT0ND6 24936626 Ki = 14 nM T52522 CFZT09 24936627 Ki = 223 nM T52522 CH7TO3 24936763 Ki = 94 nM T52522 CKD63O 24936881 Ki = 6 nM T52522 CTS43M 24936882 Ki = 20 nM T52522 CWPZ46 24936883 Ki = 259 nM T52522 C38LFU 24936885 Ki = 11 nM T52522 CL91OF 24937013 Ki = 7 nM T52522 C61SKD 24937014 Ki = 25 nM T52522 CR13DN 24937016 Ki = 961 nM T52522 CY4KV6 24937137 Ki = 165 nM T52522 CA5HY0 24937140 Ki = 93 nM T52522 CNP3A6 24937269 Ki = 18 nM T52522 C9N1UV 24937387 Ki = 517 nM T52522 CZQH42 24937389 Ki = 4.9 nM T52522 COLT89 24937390 Ki = 270 nM T52522 CX8N2G 24949262 EC50 > 1000 nM T52522 CH6YJ7 24949418 EC50 > 1000 nM T52522 CK2NO1 24949570 EC50 > 1000 nM T52522 CNV6F3 24949720 EC50 > 1000 nM T52522 C12RTH 24949722 EC50 > 1000 nM T52522 C4Q1NP 24949889 EC50 > 1000 nM T52522 CA5Q4V 24949891 EC50 > 1000 nM T52522 C1VE2O 24950053 EC50 > 1000 nM T52522 CL5CM8 24950059 EC50 > 1000 nM T52522 C8HMF4 24950061 EC50 > 1000 nM T52522 C3PB6N 24950242 EC50 > 1000 nM T52522 CEU3F6 24950403 EC50 > 1000 nM T52522 CMV2K0 24950568 EC50 > 1000 nM T52522 CL82QV 25031021 EC50 = 6.31 nM T52522 C4B0FU 25070577 IC50 = 1400 nM T52522 CB6FI3 40424734 IC50 = 8400 nM T52522 CAD31R 42611263 EC50 = 0.1585 nM T52522 C0FE1J 42625511 EC50 = 0.7943 nM T52522 C7GK2I 42625513 EC50 = 0.5012 nM T52522 CE6IF3 42625515 EC50 = 0.631 nM T52522 C1BE8M 42625517 EC50 = 0.5012 nM T52522 CL89KJ 42625587 EC50 = 1 nM T52522 CQ4O3V 42625588 EC50 = 1.585 nM T52522 C9Q0OM 42625741 EC50 = 7.943 nM T52522 CBN76E 42625743 EC50 = 25118.86 nM T52522 C6P3JN 42625821 EC50 = 1 nM T52522 C3JAT7 42625823 EC50 = 0.1995 nM T52522 C4KE6Z 42625897 EC50 = 1.259 nM T52522 C6YR7G 42625898 EC50 = 2.512 nM T52522 C8BTP0 42629372 EC50 = 7.6 nM T52522 CAJ05V 42639494 EC50 > 10000 nM T52522 C45DIE 43634116 Ki = 7890 nM T52522 CB4Q8W 44126931 EC50 > 100000 nM T52522 CWGQ16 44126933 EC50 > 100000 nM T52522 CU8M4H 44127048 EC50 > 100000 nM T52522 CXM3V6 44127050 EC50 > 100000 nM T52522 CS0B5Z 44127052 EC50 > 100000 nM T52522 C4H9TJ 44127054 EC50 > 100000 nM T52522 C2IC7Q 44127056 EC50 > 100000 nM T52522 CAW50P 44127167 EC50 > 100000 nM T52522 CJ0S7Q 44127169 EC50 > 100000 nM T52522 C53MWL 44127171 EC50 > 100000 nM T52522 CX2VJ3 44127374 EC50 > 100000 nM T52522 C8BRZ2 44127478 EC50 > 100000 nM T52522 C6XMJ7 44127479 EC50 > 100000 nM T52522 C6ULE4 44127480 EC50 > 100000 nM T52522 C1LWJ0 44127481 EC50 > 100000 nM T52522 CCI02W 44127575 EC50 > 100000 nM T52522 CL10EZ 44127677 EC50 > 100000 nM T52522 C73XYH 44127678 EC50 > 100000 nM T52522 CZ5FG8 44127679 EC50 > 100000 nM T52522 CB1W9S 44127681 EC50 > 100000 nM T52522 CY39CN 44127782 EC50 > 100000 nM T52522 C19VMJ 44186438 IC50 = 1 nM T52522 CLR40G 44219629 EC50 > 100000 nM T52522 CZ2BO8 44219630 EC50 > 100000 nM T52522 CW7D8Q 44219641 EC50 = 27 nM T52522 C27AGX 44268214 IC50 = 63 nM T52522 C9D7RS 44268249 IC50 = 10 nM T52522 C5E2MI 44268254 IC50 = 500 nM T52522 CAY8L6 44268264 EC50 = 5 nM T52522 CNQ7X8 44268266 IC50 = 84 nM T52522 C72KSE 44268267 EC50 = 30 nM T52522 CLR0X8 44268268 IC50 = 240 nM T52522 C9TB2F 44268273 IC50 = 100 nM T52522 C6NY3M 44268274 IC50 = 370 nM T52522 CGJT32 44268275 IC50 = 130 nM T52522 CZ3W8B 44268277 IC50 = 58 nM T52522 CLS1U8 44268281 IC50 = 250 nM T52522 C6R8SP 44268295 IC50 = 500 nM T52522 C0UG8A 44268305 IC50 = 20 nM T52522 C2AJI5 44268308 IC50 = 190 nM T52522 CY6X8E 44268320 IC50 = 170 nM T52522 CCH34M 44268322 IC50 = 150 nM T52522 CAD4P0 44268324 IC50 = 280 nM T52522 CI91WY 44268327 IC50 = 3000 nM T52522 CMU89C 44268341 IC50 = 630 nM T52522 CS87PI 44268349 IC50 = 21 nM T52522 CB7F6R 44268352 IC50 = 220 nM T52522 CPNS03 44268358 IC50 = 3000 nM T52522 C9JZ5T 44268365 IC50 = 230 nM T52522 CP2G7C 44268367 IC50 = 11 nM T52522 C1S3AB 44268464 IC50 = 110 nM T52522 C29IOC 44268470 IC50 = 230 nM T52522 CI64OC 44268478 IC50 = 110 nM T52522 CU84BM 44268479 IC50 = 210 nM T52522 CQY09P 44268482 IC50 = 2000 nM T52522 CRV1T3 44268495 IC50 = 170 nM T52522 CU21DW 44268496 IC50 = 700 nM T52522 CWG2Q7 44268498 IC50 = 120 nM T52522 C4D1OQ 44268509 IC50 = 220 nM T52522 C3YGB4 44268520 IC50 = 130 nM T52522 C5TZ8J 44268534 IC50 = 400 nM T52522 CS73JY 44268539 IC50 = 450 nM T52522 CN8P2B 44268556 IC50 = 430 nM T52522 CES3Y9 44268563 IC50 = 230 nM T52522 CY5J3N 44268568 IC50 = 350 nM T52522 CREN46 44268569 IC50 = 290 nM T52522 C0BR2A 44268570 IC50 = 720 nM T52522 C9H1IF 44268571 IC50 = 5000 nM T52522 CBZ7N6 44268572 IC50 = 1000 nM T52522 C2LYD1 44268604 IC50 = 200 nM T52522 CD7UZ0 44268605 IC50 = 540 nM T52522 CF3VU1 44268632 IC50 = 400 nM T52522 CW7A6K 44280795 IC50 = 8500 nM T52522 CR8D7Y 44280858 IC50 = 2500 nM T52522 C4JLV9 44280860 IC50 = 6500 nM T52522 C49FOW 44280903 IC50 = 1500 nM T52522 CM6C4J 44280904 IC50 = 4500 nM T52522 CJ1B9Z 44280957 IC50 = 51000 nM T52522 CM9R8D 44281037 IC50 = 10000 nM T52522 CPO25L 44281073 IC50 = 24000 nM T52522 CI4NE5 44281074 IC50 = 12000 nM T52522 CG7A5O 44281097 IC50 = 3500 nM T52522 CS84VC 44281218 IC50 = 1500 nM T52522 CIPT87 44281219 IC50 = 2000 nM T52522 C1S3HD 44281255 IC50 = 5500 nM T52522 CZT1Q6 44281276 IC50 = 1000 nM T52522 COB42G 44281277 IC50 = 1415 nM T52522 C28KLB 44281344 IC50 = 9500 nM T52522 C65JLA 44281371 IC50 = 5000 nM T52522 CD78QG 44281372 IC50 = 90000 nM T52522 CBNZ27 44281384 IC50 = 5000 nM T52522 CG3D5J 44281395 IC50 = 2500 nM T52522 CBL4F1 44281396 IC50 = 490 nM T52522 CO9F8Q 44281400 IC50 = 1430 nM T52522 CT0XW9 44281407 IC50 = 2500 nM T52522 CK3Z4L 44281408 IC50 = 5400 nM T52522 C7P3WY 44281424 IC50 = 15000 nM T52522 CIO1V4 44281425 IC50 = 5000 nM T52522 CJU5O2 44281467 IC50 = 3000 nM T52522 CI1C5Q 44281468 IC50 = 2000 nM T52522 CTL1G7 44281469 IC50 = 695 nM T52522 CEN7H9 44281470 IC50 = 2500 nM T52522 CC90RN 44281530 IC50 = 720 nM T52522 CLXI95 44281531 IC50 = 9500 nM T52522 C0DG5M 44285225 IC50 = 1000 nM T52522 CNO3I4 44285226 IC50 = 1200 nM T52522 C7L5MN 44285529 IC50 = 4000 nM T52522 CUF3O2 44285634 IC50 = 270 nM T52522 CTIA64 44285685 IC50 = 3000 nM T52522 C0JY4C 44285692 IC50 = 30000 nM T52522 CPQ16U 44286964 Ki = 39700 nM T52522 CKL84D 44286965 Ki = 260 nM T52522 C2IJ9G 44286980 Ki = 73700 nM T52522 CPN74V 44286983 Ki = 170 nM T52522 CE5GK6 44287268 Ki = 42600 nM T52522 CD0E2S 44287321 Ki = 17100 nM T52522 CA72HF 44287337 Ki = 112 nM T52522 C53RQT 44298256 IC50 = 52 nM T52522 C5EXK1 44298281 IC50 = 8000 nM T52522 C82TAV 44298288 IC50 = 510 nM T52522 C0ICR9 44298290 IC50 = 750 nM T52522 COTF72 44298306 IC50 = 2500 nM T52522 CX4QG5 44298314 IC50 = 42 nM T52522 CIJ6H2 44298315 IC50 = 100 nM T52522 CDCP96 44298497 IC50 = 530 nM T52522 CNK60M 44298515 IC50 = 620 nM T52522 CZHU81 44298516 IC50 = 900 nM T52522 CJ1X0Z 44298533 IC50 = 1300 nM T52522 CRD69E 44298695 IC50 = 1000 nM T52522 CP72DS 44298700 IC50 = 7000 nM T52522 CSKD26 44298718 IC50 = 2000 nM T52522 CBW06V 44298728 IC50 = 36000 nM T52522 CVN75C 44298731 IC50 = 630 nM T52522 C67YCD 44298752 IC50 = 6500 nM T52522 CO9BE8 44298761 IC50 = 7300 nM T52522 CYGM23 44298767 IC50 = 10000 nM T52522 CD51GN 44298769 IC50 = 440 nM T52522 CE01UQ 44298781 IC50 = 1000 nM T52522 CUK01S 44298787 IC50 = 340 nM T52522 CFRN96 44298821 IC50 = 180 nM T52522 C40OYU 44298822 IC50 = 7500 nM T52522 C19XHR 44298823 IC50 = 1500 nM T52522 CSW8G0 44298843 IC50 = 240 nM T52522 CQID30 44298849 IC50 = 460 nM T52522 C8FL6R 44298850 IC50 = 450 nM T52522 CHJR57 44298851 IC50 = 63 nM T52522 C2GBS7 44298852 IC50 = 140 nM T52522 C6GD9N 44301617 IC50 = 90000 nM T52522 CI0OY1 44301618 IC50 = 1900 nM T52522 C4P1OD 44301764 IC50 = 620 nM T52522 CCH74I 44301803 IC50 = 2500 nM T52522 C3T9OF 44301804 IC50 = 4000 nM T52522 CY63AQ 44301805 IC50 = 3000 nM T52522 CA3VZ2 44301806 IC50 = 8000 nM T52522 C2OJ3N 44301818 IC50 = 5700 nM T52522 CNZ68T 44301819 IC50 = 2000 nM T52522 CMFW56 44301831 IC50 = 3000 nM T52522 CJB9L8 44301832 IC50 = 3000 nM T52522 C4DZ6V 44301842 IC50 = 6300 nM T52522 CW02XN 44301843 IC50 = 910 nM T52522 C6P8UW 44301866 IC50 = 1000 nM T52522 C8T7OB 44301867 IC50 = 2100 nM T52522 CS4ET3 44301880 IC50 = 49000 nM T52522 CM4G9Z 44301881 IC50 = 93000 nM T52522 C6VDZ8 44301886 IC50 = 16000 nM T52522 C08SKL 44301979 IC50 = 47000 nM T52522 C8EGA1 44302005 IC50 = 50000 nM T52522 C9J6RY 44303192 IC50 = 7000 nM T52522 CN0DE9 44303198 IC50 = 28 nM T52522 CA4BQ1 44306956 IC50 = 360 nM T52522 C70GLV 44306959 IC50 = 380 nM T52522 C9HL3E 44306979 IC50 = 990 nM T52522 C75OJI 44306985 IC50 = 1000 nM T52522 CH58SX 44306991 IC50 = 1300 nM T52522 C0XI5A 44306992 IC50 = 630 nM T52522 CN23SP 44307007 IC50 = 410 nM T52522 C4LRJ3 44307063 IC50 = 230 nM T52522 CYI2V9 44307064 IC50 = 430 nM T52522 C7KWF2 44307065 IC50 = 900 nM T52522 C3H9QV 44307113 IC50 = 50 nM T52522 CC4IL0 44307144 IC50 = 430 nM T52522 CK0WG5 44307166 IC50 = 100 nM T52522 CLB56U 44307186 IC50 = 94 nM T52522 CYX08L 44307196 IC50 = 380 nM T52522 CNCV21 44307205 IC50 = 640 nM T52522 C5Q4MP 44307333 IC50 = 620 nM T52522 CVK8S0 44307340 IC50 = 110 nM T52522 C1RYI9 44307343 IC50 = 520 nM T52522 CK1P5Z 44307378 IC50 = 490 nM T52522 CV1Z0F 44307379 IC50 = 750 nM T52522 C5NIP7 44307396 IC50 = 150 nM T52522 C9G4UO 44309272 EC50 = 920 nM T52522 CKWA37 44309523 EC50 = 920 nM T52522 CMJX34 44309649 EC50 > 100000 nM T52522 CFHD64 44312269 Ki = 13900 nM T52522 CVX04Z 44312421 Ki = 150 nM T52522 CF3H5U 44312924 IC50 = 760 nM T52522 CY4K0A 44312949 IC50 = 300 nM T52522 C3L4PJ 44313090 IC50 = 300 nM T52522 CL2UV6 44313150 IC50 = 710 nM T52522 CPA5B7 44313161 IC50 = 990 nM T52522 C15EMW 44328703 Ki = 12 nM T52522 CV8J4A 44331302 EC50 = 30 nM T52522 C97IJY 44331346 EC50 = 30 nM T52522 C0RDZ3 44331351 EC50 = 20000 nM T52522 CIFO93 44331425 EC50 = 1000 nM T52522 C5Y8GN 44331426 EC50 = 5 nM T52522 CU4EQ5 44331443 EC50 = 20 nM T52522 CWE69G 44331444 EC50 = 12 nM T52522 CI17GW 44331766 EC50 > 1000 nM T52522 CR36NA 44335496 IC50 = 10000 nM T52522 C5BX2N 44335497 IC50 = 8000 nM T52522 CD7ZV4 44335498 IC50 = 1000 nM T52522 C9UE7G 44335499 IC50 = 6000 nM T52522 CDS5L1 44335534 IC50 = 200 nM T52522 C7MC1U 44335548 IC50 = 410 nM T52522 CY7LH9 44335560 IC50 = 8000 nM T52522 C6IA8P 44335562 IC50 = 2000 nM T52522 CLE91U 44335572 IC50 = 5000 nM T52522 C4B8OE 44335588 IC50 = 9000 nM T52522 C7A4UT 44335603 IC50 = 10000 nM T52522 CFX90I 44335618 IC50 = 8000 nM T52522 C14ILU 44335628 IC50 = 10000 nM T52522 CX8QZ4 44335651 IC50 = 10000 nM T52522 C03GDI 44335663 IC50 = 820 nM T52522 CL2BX0 44335833 IC50 = 1000 nM T52522 C4M8EN 44335844 IC50 = 50000 nM T52522 C3DP9K 44335882 IC50 = 8000 nM T52522 CA6X9Y 44339091 EC50 = 1.585 nM T52522 CTBA45 44339100 EC50 > 1000 nM T52522 C4PU1O 44349588 IC50 = 260 nM T52522 CS1L9V 44349629 IC50 = 50 nM T52522 CO27RQ 44349645 IC50 = 710 nM T52522 C6WP1E 44349646 IC50 = 66 nM T52522 CZK46C 44369602 EC50 = 50.12 nM T52522 C3M7BC 44377315 IC50 = 1000 nM T52522 CS6C8L 44377316 IC50 = 1000 nM T52522 CI1MN9 44377412 IC50 = 10000 nM T52522 CEW6J9 44377513 IC50 = 2000 nM T52522 C8DYK5 44377514 IC50 = 730 nM T52522 CRB49F 44377517 IC50 = 5000 nM T52522 C3XLD1 44377636 IC50 = 3500 nM T52522 C3BQ1X 44377637 IC50 = 2000 nM T52522 CHB6Q2 44377650 IC50 = 5000 nM T52522 CNEO30 44377665 IC50 = 50000 nM T52522 CKI9O8 44377677 IC50 = 2000 nM T52522 CQEA58 44377687 IC50 = 1000 nM T52522 C49FSC 44377753 IC50 = 13000 nM T52522 CW42ZY 44377754 IC50 = 760 nM T52522 C04XMY 44377755 IC50 = 10000 nM T52522 C02ZPF 44377957 IC50 = 5300 nM T52522 CG2F6I 44386630 Ki = 7.2 nM T52522 C7DT6S 44391257 Ki = 0.631 nM T52522 C0UEV5 44391270 Ki = 1000 nM T52522 C0CBD4 44392457 EC50 = 10 nM T52522 CES46V 44392480 EC50 = 11 nM T52522 CXO92R 44392490 EC50 = 69 nM T52522 CHIC83 44392508 EC50 = 46 nM T52522 C7D8AU 44392519 EC50 = 16 nM T52522 CMH6N4 44392534 EC50 = 2.2 nM T52522 C7QJN5 44392542 EC50 = 7.6 nM T52522 CND67K 44392552 EC50 = 19 nM T52522 CS3H7D 44392558 EC50 = 36 nM T52522 CCZQ48 44392566 EC50 = 1.5 nM T52522 C83OKR 44392575 EC50 = 9.6 nM T52522 CADQ67 44392577 EC50 = 18 nM T52522 CGI3O1 44393827 Ki = 35.4 nM T52522 C8OFH5 44393865 Ki = 5.9 nM T52522 C5H0IF 44393894 Ki = 7.8 nM T52522 CE9CQ1 44393937 Ki = 8.5 nM T52522 CL7DP2 44393971 Ki = 11.6 nM T52522 CI4J7L 44396488 EC50 = 6.8 nM T52522 CY46LP 44396509 EC50 = 12 nM T52522 CB37RE 44396513 EC50 = 6.2 nM T52522 CE1MS4 44396530 EC50 = 7.3 nM T52522 C2YP6O 44396531 EC50 = 5.6 nM T52522 CLYG39 44396532 EC50 = 21 nM T52522 CJ75RF 44396559 EC50 = 7.7 nM T52522 CN7HX8 44396568 EC50 = 19 nM T52522 C2DOA1 44396577 EC50 = 6.6 nM T52522 CHXA19 44396596 EC50 = 6.6 nM T52522 CZ71YN 44396659 Ki = 223 nM T52522 CW4OR6 44396715 EC50 = 1.3 nM T52522 C4BXY6 44396729 Ki = 70 nM T52522 CRY62C 44396736 EC50 = 1.2 nM T52522 C4WO2Y 44396737 EC50 = 7.2 nM T52522 C6CZX4 44396738 EC50 = 60 nM T52522 CUO7X8 44396779 EC50 = 3.1 nM T52522 C53GBI 44396798 EC50 = 13 nM T52522 C0EXA1 44407083 IC50 > 10000 nM T52522 CSA2X5 44419254 EC50 = 2.4 nM T52522 CG5XU6 44419315 EC50 > 10000 nM T52522 C4ABS0 44419316 EC50 > 10000 nM T52522 CQ89AE 44419324 EC50 > 10000 nM T52522 CFG74O 44419332 EC50 > 10000 nM T52522 C5YBA0 44423639 Ki > 100000 nM T52522 C3XR8N 44423640 Ki = 13.9 nM T52522 C45ISV 44423641 Ki = 501 nM T52522 CK1XO7 44423643 Ki = 2.82 nM T52522 CD72TX 44423644 Ki = 81.4 nM T52522 C34MXL 44423645 Ki = 15.5 nM T52522 C7IAO1 44423646 Ki = 458 nM T52522 CD5JR4 44424578 Ki = 9280 nM T52522 CI8X5A 44424579 Ki = 31400 nM T52522 C6YT8M 44424580 Ki > 100000 nM T52522 C2AE3K 44424581 Ki = 56234.13 nM T52522 CR9LT6 44425580 EC50 = 0.096 nM T52522 C5P4OW 44433250 Ki = 6.63 nM T52522 C6MCP3 44434116 EC50 = 0.706 nM T52522 C53QID 44434117 EC50 = 2.55 nM T52522 CID6M7 44434125 EC50 = 0.049 nM T52522 CGW3H6 44434126 EC50 = 0.038 nM T52522 C7E5DW 44434127 EC50 = 0.053 nM T52522 C0YJ5E 44434128 EC50 = 0.164 nM T52522 CTR6H9 44434130 EC50 = 0.022 nM T52522 CN8G6D 44441226 EC50 = 100 nM T52522 C4Q1JB 44441227 EC50 = 125.89 nM T52522 CC34NU 44441228 EC50 = 50.12 nM T52522 CE34HD 44441229 EC50 = 158.49 nM T52522 CXE23W 44441230 EC50 = 50.12 nM T52522 CZ96SJ 44441231 EC50 = 100 nM T52522 CTWM30 44441232 EC50 = 398.11 nM T52522 CA8E5H 44441233 EC50 = 316.23 nM T52522 CP2H0M 44441234 EC50 = 79.43 nM T52522 CZ2K7C 44441235 EC50 = 630.96 nM T52522 CR9B1F 44441236 EC50 = 5011.87 nM T52522 C6MFP8 44444153 EC50 > 10000 nM T52522 C1QZW9 44444154 EC50 > 10000 nM T52522 CGDZ68 44444166 EC50 > 10000 nM T52522 C9OIT6 44444167 EC50 > 10000 nM T52522 CG2QI4 44444169 EC50 > 10000 nM T52522 C58UHL 44444170 Ki = 2700 nM T52522 CUAN40 44444171 EC50 > 10000 nM T52522 CVQ59T 44444172 EC50 > 10000 nM T52522 C60YDC 44444173 EC50 = 35.2 nM T52522 C1IB7H 44444175 EC50 > 10000 nM T52522 CZ0VJ5 44444176 EC50 > 10000 nM T52522 CD74SN 44444179 Ki = 38 nM T52522 C5TM3W 44444185 Ki = 390 nM T52522 C16XQT 44444187 Ki = 280 nM T52522 C6PS3A 44444188 Ki = 200 nM T52522 CZAK23 44444189 Ki = 71 nM T52522 C9A3KP 44444191 Ki = 57 nM T52522 CA08VR 44444193 Ki = 26 nM T52522 CNS8K2 44444195 Ki = 120 nM T52522 C9C1PF 44446497 IC50 = 777000 nM T52522 CN9BV2 44446499 IC50 = 820000 nM T52522 C12XGE 44456400 Ki > 10000 nM T52522 C1A6ZC 44457929 IC50 = 570 nM T52522 C7O0IE 44458134 IC50 = 3300 nM T52522 C68NOT 44461468 IC50 = 3000 nM T52522 CDZ56W 44461485 IC50 = 8500 nM T52522 CM5ZH4 44461486 IC50 = 4500 nM T52522 C2GZ3R 44461488 IC50 = 100000 nM T52522 C1L6GN 44461489 IC50 = 6500 nM T52522 CQ8UE4 44461716 IC50 = 7000 nM T52522 C4TMP7 44461717 IC50 = 7000 nM T52522 C39FRG 44461718 IC50 = 330 nM T52522 CM4F7J 44461719 IC50 = 9000 nM T52522 C4DL5C 44469677 IC50 > 10000 nM T52522 C2QK4J 44472590 IC50 > 20000 nM T52522 CQ8C3F 44472591 IC50 = 2200 nM T52522 CC2TA5 44472592 IC50 > 20000 nM T52522 CWN95E 44472610 IC50 > 20000 nM T52522 C1H2ZT 44472612 IC50 > 20000 nM T52522 C9G5ID 44472613 IC50 > 20000 nM T52522 C5N4KE 44472633 IC50 > 20000 nM T52522 CEH82X 44472636 IC50 > 20000 nM T52522 CMH3J4 44472637 IC50 > 20000 nM T52522 CC6G0Z 44517692 EC50 = 20 nM T52522 C5BYX7 44517694 EC50 = 20 nM T52522 CY8PO3 44517696 EC50 = 20 nM T52522 CV92IJ 44541354 IC50 > 30 nM T52522 C1E3MT 44554514 EC50 = 13 nM T52522 CE18ZY 44560791 EC50 > 1000 nM T52522 C7V8EF 44560792 EC50 > 1000 nM T52522 CMP8T6 44560793 EC50 > 1000 nM T52522 CAF8L7 44565931 EC50 = 290 nM T52522 CDUZ13 44565932 EC50 = 1200 nM T52522 CBD52U 44574651 EC50 > 100000 nM T52522 CSGI84 44574685 EC50 > 100000 nM T52522 CIF02K 44574686 EC50 > 100000 nM T52522 C4PN5S 44574687 EC50 > 100000 nM T52522 C6BVQ7 44574688 EC50 > 100000 nM T52522 C6UTI8 44574720 EC50 > 100000 nM T52522 C0RB7H 44574721 EC50 > 100000 nM T52522 C56UZO 44574722 EC50 > 100000 nM T52522 CVP31K 44574723 EC50 > 100000 nM T52522 CM53PL 44574757 EC50 > 100000 nM T52522 CLG2N1 44574758 EC50 > 100000 nM T52522 C6E2SN 44574759 EC50 > 100000 nM T52522 CIS5B4 44574825 EC50 > 100000 nM T52522 CK2H8G 44574826 EC50 > 100000 nM T52522 CU7H5I 44574827 EC50 > 100000 nM T52522 C9GZ3R 44574867 EC50 > 100000 nM T52522 CL7SJ3 44574868 EC50 > 100000 nM T52522 C9HE8U 44574913 EC50 > 100000 nM T52522 CO3V6F 44574978 EC50 > 100000 nM T52522 C5NS6H 44581972 Ki = 2290.87 nM T52522 CK8Z1P 44581973 Ki = 2398.83 nM T52522 C3UQ9Z 44581974 Ki > 6309.57 nM T52522 C3L5ER 44583033 IC50 = 0.0013 nM T52522 CXD63G 44589133 EC50 = 1156 nM T52522 CS08ED 44589400 EC50 = 5895 nM T52522 CJ0D9X 44591506 EC50 > 1000 nM T52522 C32HSU 44591507 EC50 = 3200 nM T52522 CWQ2K4 44591508 EC50 = 1100 nM T52522 C5KTS1 44609903 EC50 = 14 nM T52522 CH2Z3O 44610056 EC50 = 20.9 nM T52522 C9G8WB 44610361 EC50 = 116 nM T52522 CO3I5F 44622849 Ki = 7600 nM T52522 CC18SZ 45101519 EC50 = 1 nM T52522 CL9UT7 45101520 EC50 = 1.2 nM T52522 C04EWA 45101521 EC50 = 5.4 nM T52522 CWIL37 45101522 EC50 = 1.8 nM T52522 C7CM3S 45101537 EC50 > 10000 nM T52522 C07LMT 45267257 EC50 = 10 nM T52522 C5P2KR 45268128 EC50 = 30 nM T52522 C7NC2T 45268136 EC50 = 30 nM T52522 C7GPS1 45269025 EC50 = 10 nM T52522 C43UZN 45270690 EC50 = 20 nM T52522 CCZ10H 45270697 EC50 = 10 nM T52522 CK48MV 45271517 EC50 = 20 nM T52522 C13VYN 45271518 EC50 = 10 nM T52522 CMU01B 45271523 EC50 = 10 nM T52522 CS27QE 45272430 EC50 = 10 nM T52522 CL76SG 45272431 EC50 = 10 nM T52522 C6GW4V 45273276 EC50 = 30 nM T52522 CH10SC 45273280 EC50 = 30 nM T52522 CPJB52 45280075 EC50 > 10000 nM T52522 CZEB18 45375919 EC50 = 2.9 nM T52522 C6QES8 45380471 EC50 > 10000 nM T52522 CZ73IE 45381852 EC50 > 10000 nM T52522 CNI72R 45381932 EC50 > 10000 nM T52522 C7RYF5 45483810 EC50 = 0.2 nM T52522 C70MIX 45483813 EC50 = 0.1 nM T52522 C6IU9K 45483814 EC50 = 0.7 nM T52522 CJ5LO8 45483815 EC50 = 2.8 nM T52522 C1W0IA 45483816 EC50 = 0.4 nM T52522 CKY85H 45483825 EC50 = 70 nM T52522 CVI32P 45483830 EC50 = 20 nM T52522 CI96VQ 45483831 EC50 = 170 nM T52522 CNX06B 45483838 EC50 = 131 nM T52522 CBN09R 45483839 EC50 > 10000 nM T52522 CC3F7O 45483843 EC50 = 0.6 nM T52522 CH1BC2 45483844 EC50 = 1.5 nM T52522 CAZ4C7 45483846 EC50 = 13.4 nM T52522 CEH1G2 45483847 EC50 = 1.7 nM T52522 C4ISE8 45483848 EC50 > 10000 nM T52522 CGD86T 45483849 EC50 > 10000 nM T52522 CSQT68 45483852 EC50 = 0.5 nM T52522 CN1KI6 45483864 EC50 = 0.4 nM T52522 C43ETK 45483868 EC50 = 0.6 nM T52522 C9QR8M 45484536 EC50 = 0.9 nM T52522 CN2L9F 45484537 EC50 = 11.6 nM T52522 C4JH6P 45484558 EC50 = 4.1 nM T52522 CS5RA6 45484568 EC50 = 0.5 nM T52522 C8YBJ6 45484569 EC50 = 1.2 nM T52522 CHQ83C 45484583 EC50 = 1.1 nM T52522 CQ07ZN 45484584 EC50 = 1 nM T52522 CI0M5N 45484646 EC50 = 9 nM T52522 C05PBD 46176231 IC50 > 10000 nM T52522 CWK38C 46221395 EC50 = 5 nM T52522 CJYX12 46221396 EC50 = 39 nM T52522 CW6C3U 46221397 EC50 = 14 nM T52522 C2Q6PE 46221398 EC50 = 25 nM T52522 CN9MC4 46221603 EC50 = 18 nM T52522 CRU86Y 46221604 EC50 = 115 nM T52522 C4U3XI 46232768 EC50 = 2.4 nM T52522 CI35QZ 46232769 EC50 = 0.7 nM T52522 C1TS7M 46232815 EC50 = 5167 nM T52522 CE79ZN 46232816 EC50 = 68 nM T52522 CAF43W 46232856 EC50 = 3.4 nM T52522 CW1M4Q 46232857 EC50 = 11.9 nM T52522 CO2B9C 46232973 EC50 = 1.4 nM T52522 CF1B6A 46232974 EC50 = 97.7 nM T52522 CSNR69 46233013 EC50 = 14.3 nM T52522 C7NA1H 46832227 EC50 = 2511.89 nM T52522 CNA42V 46832232 EC50 = 0.1259 nM T52522 CN7MG5 46832505 EC50 = 2.512 nM T52522 CJ5B4A 46832507 EC50 = 1.585 nM T52522 CW0JV6 46832509 EC50 = 0.2512 nM T52522 C7TN0H 46832510 EC50 = 0.3981 nM T52522 C04XPW 46832798 EC50 = 0.3981 nM T52522 CF72EA 46832801 EC50 = 2.512 nM T52522 CUTY31 46832803 EC50 = 2.512 nM T52522 CQ1BJ4 46832804 EC50 = 1.995 nM T52522 C6VS1A 46833102 EC50 = 1.585 nM T52522 CSYQ43 46833103 EC50 = 7.943 nM T52522 CQ3TM8 46845697 IC50 > 20000 nM T52522 CJV15G 46845698 IC50 = 15000 nM T52522 C0DB5H 46845699 IC50 = 16000 nM T52522 C2D6ZI 46881527 IC50 > 20000 nM T52522 CIP0H2 46881528 IC50 > 20000 nM T52522 CZ0PU9 46881529 IC50 > 10000 nM T52522 CTV6U8 46881530 IC50 = 6000 nM T52522 CFA38Z 46881531 IC50 > 10000 nM T52522 CIJU02 46881573 IC50 = 15000 nM T52522 C4YNT0 46881574 IC50 > 10000 nM T52522 CV5R2L 46881575 IC50 = 13000 nM T52522 CULH08 46881576 IC50 = 1100 nM T52522 CYLF92 46881614 IC50 > 20000 nM T52522 CT56SD 46881615 IC50 > 20000 nM T52522 CLB86Z 46881616 IC50 > 10000 nM T52522 CJ1VO4 46881617 IC50 = 8700 nM T52522 C6D5IZ 46881618 IC50 = 1700 nM T52522 CTC02J 46881650 IC50 > 10000 nM T52522 CN9TK8 46881651 IC50 = 1700 nM T52522 CWZ4H5 46881652 IC50 > 10000 nM T52522 CZQ6C8 46881653 IC50 > 20000 nM T52522 CD27OS 46881698 IC50 = 6700 nM T52522 CGP45C 46881699 IC50 > 10000 nM T52522 C7BPN3 46881700 IC50 > 10000 nM T52522 CMR6C9 46881701 IC50 = 7800 nM T52522 C8QS6V 46881750 IC50 = 1100 nM T52522 C8XST7 46881751 IC50 > 20000 nM T52522 CW60AO 46881752 IC50 > 10000 nM T52522 CFIE98 46881753 IC50 > 20000 nM T52522 C4EOF8 46881796 IC50 = 600 nM T52522 C9HO2J 46881797 IC50 > 20000 nM T52522 CX8ZS6 46881798 IC50 > 20000 nM T52522 C9OE3N 46881799 IC50 > 20000 nM T52522 CV75XD 46881838 IC50 > 20000 nM T52522 CVR9M2 46881839 IC50 = 3600 nM T52522 C4D1XF 46881840 IC50 > 20000 nM T52522 CK0N6A 46881869 IC50 > 20000 nM T52522 C9CUP4 46881870 IC50 > 20000 nM T52522 C53CIB 46881871 IC50 > 20000 nM T52522 CGZ7K5 46881872 IC50 = 16000 nM T52522 CHJ9D1 46881899 IC50 > 20000 nM T52522 C4D7PW 46881900 IC50 = 400 nM T52522 CI7Q6U 46881901 IC50 = 60 nM T52522 CTX8N0 46881902 IC50 = 5300 nM T52522 CR1H5N 46881935 IC50 > 10000 nM T52522 CQ87KZ 46881936 IC50 > 10000 nM T52522 CKDO83 46881937 IC50 > 20000 nM T52522 C7W1LE 46881938 IC50 = 3000 nM T52522 CXDJ80 46881980 IC50 > 20000 nM T52522 CP5O9V 46881981 IC50 = 6900 nM T52522 C4N0KV 46881982 IC50 = 1700 nM T52522 C50CFL 46881983 IC50 > 10000 nM T52522 C50GNW 46882028 IC50 = 4700 nM T52522 CBC6Z5 46882029 IC50 = 600 nM T52522 C2Y3DO 46882030 IC50 = 400 nM T52522 CWG7Z8 46882031 IC50 = 400 nM T52522 CWI86A 46882084 IC50 = 100 nM T52522 CSG57M 46887146 Ki > 10000 nM T52522 CBN3V6 46889642 Ki = 1260 nM T52522 CG72PB 46889643 Ki = 120 nM T52522 C8S4LM 46889670 Ki = 3 nM T52522 CEF90S 46889699 Ki = 40 nM T52522 CH4Z0F 46889700 Ki = 13 nM T52522 C8K6HX 46889701 Ki = 135 nM T52522 CAO57K 46889727 Ki = 78 nM T52522 CTP3E7 46889728 Ki = 38 nM T52522 CW9LS6 46889729 Ki = 50 nM T52522 C7RI4K 46889730 Ki = 17 nM T52522 C4ISX8 46889767 Ki = 80 nM T52522 C3ZY5J 46889768 Ki = 9 nM T52522 C3F4IQ 46889769 Ki = 2.4 nM T52522 C1P5WV 46889770 Ki = 17 nM T52522 C02HNI 46889771 Ki = 37 nM T52522 C4D5FH 46889772 Ki = 8 nM T52522 CKIM07 46889809 Ki = 57 nM T52522 C6CY1S 46889810 Ki = 0.5 nM T52522 C26WTA 46889811 Ki = 0.2 nM T52522 C2GC4K 46889812 Ki = 0.1 nM T52522 C9P4TD 46889852 Ki = 0.2 nM T52522 C1YVO4 46889853 Ki = 0.2 nM T52522 CFY40T 46889854 Ki = 0.3 nM T52522 CV5N9U 46938906 EC50 = 0.37 nM T52522 C15ZGJ 46938907 EC50 = 0.13 nM T52522 CK8V2H 49800025 EC50 = 0.5012 nM T52522 CV5G1H 49861320 EC50 = 50 nM T52522 C6OQV2 49862237 Ki > 1000 nM T52522 CX5TY8 49864332 Ki = 24.7 nM T52522 C3GAQ5 49864333 Ki = 1 nM T52522 CN9R1Z 49864334 Ki = 25.1 nM T52522 CP6XL8 49864335 Ki = 1.9 nM T52522 CCO9X4 49864355 Ki = 26.5 nM T52522 CO4BD7 49864356 Ki = 1.8 nM T52522 C5KHJ2 49864357 Ki = 19.8 nM T52522 C9NOK6 49864358 Ki = 1.2 nM T52522 CY0FL3 49864377 Ki = 9.4 nM T52522 CN87YW 49864378 Ki = 30.2 nM T52522 CEQI63 49864379 Ki = 1.8 nM T52522 CJ04XU 49864380 Ki = 2.7 nM T52522 CD48CK 49864381 Ki = 48.9 nM T52522 C7MZC6 49864394 Ki = 11.8 nM T52522 C7C8PK 49864395 EC50 = 0.03162 nM T52522 C5O7HP 49864396 Ki = 0.6 nM T52522 CLK3Y5 49864397 Ki = 0.8 nM T52522 C87HDG 49864412 Ki = 7.2 nM T52522 C8KVZ6 49864413 Ki = 362 nM T52522 CUR2Z4 49864414 Ki = 40.4 nM T52522 CVA6H4 49864415 Ki = 3.8 nM T52522 C8U7ID 49864416 Ki = 4 nM T52522 CFA63G 49864439 Ki = 151 nM T52522 CQVR67 49864440 Ki = 6.3 nM T52522 CZV9N8 49864441 Ki = 4.4 nM T52522 C62FLG 49864442 Ki = 0.3 nM T52522 CJQI64 49864443 Ki > 1000 nM T52522 C6SL3T 49864460 Ki = 3 nM T52522 C1WL8J 49864461 Ki = 18.3 nM T52522 C2RY0J 50878551 Ki > 10000 nM T52522 C1W6TV 50898777 Ki > 10000 nM T52522 CXMZ73 50898778 Ki > 10000 nM T52522 CLY9W1 50994950 IC50 = 10900 nM T52522 C2CH1R 50995330 IC50 = 5200 nM T52522 CE4KP1 51050257 Ki > 10000 nM T52522 CYR21W 51346867 IC50 = 2509 nM T52522 C4Z2FY 51347436 IC50 > 20000 nM T52522 CQG7X2 51349173 EC50 > 10000 nM T52522 C1F0DX 52941476 Ki = 10 nM T52522 CZMS46 52941603 Ki = 135 nM T52522 C83BMV 52943362 Ki = 4 nM T52522 C3B2OF 52943383 Ki = 68 nM T52522 C61ZLX 52943770 Ki = 873 nM T52522 CE13YX 52943919 Ki = 6 nM T52522 C5TW1N 52943932 Ki = 42 nM T52522 CVE5Q9 52943968 Ki = 139 nM T52522 C69LKY 52943969 Ki = 117 nM T52522 CP6U9S 52944986 Ki = 25 nM T52522 C0TWA8 52946357 Ki = 440 nM T52522 CFX1D5 52946430 Ki = 370 nM T52522 CI2PT6 52946537 Ki = 14 nM T52522 C7ULQ8 52947060 Ki = 100 nM T52522 CHK30N 52947443 Ki = 30 nM T52522 CD7EW1 52947562 Ki = 189 nM T52522 CED37H 52948056 Ki = 19 nM T52522 CN0F9Z 52948612 Ki > 10000 nM T52522 C04PTF 52948728 Ki = 589 nM T52522 C6E9TK 52948792 Ki = 88 nM T52522 CU1R7B 52948805 Ki = 10 nM T52522 CI7S6O 52949488 Ki = 11 nM T52522 CMX86D 52949489 Ki = 30 nM T52522 C9VYT6 52949934 Ki = 80 nM T52522 CR3XD8 53239456 EC50 = 2.4 nM T52522 CUE05Y 53307431 EC50 = 125.89 nM T52522 CP0LN7 53307432 EC50 = 1.585 nM T52522 C57DOH 53318280 IC50 = 780 nM T52522 CX1G3F 53318455 EC50 = 1.3 nM T52522 CJAH78 53319639 IC50 = 2790 nM T52522 C3S1ZO 53319788 EC50 = 3.3 nM T52522 CA45EM 53326195 IC50 = 2180 nM T52522 C9SDC2 53326196 IC50 = 3530 nM T52522 CM5WF2 53326197 IC50 = 297 nM T52522 CNS26Q 53326837 EC50 = 0.9 nM T52522 C3EAT2 53326839 IC50 = 3530 nM T52522 CLN6B9 53357711 EC50 = 1 nM T52522 CL7US4 53357712 EC50 = 0.7943 nM T52522 CO47UB 53379897 EC50 = 0.4 nM T52522 COT06P 53380558 EC50 = 3.9 nM T52522 CK1MZ6 53380559 EC50 = 2.8 nM T52522 C7WKR1 53387673 Ki > 10000 nM T52522 CFB1N5 53387674 Ki > 10000 nM T52522 C9GXQ3 53495160 IC50 = 11 nM T52522 CGLI46 54417230 IC50 = 50118.72 nM T52522 C3KRU5 54580128 EC50 = 17 nM T52522 CFNI73 54580129 EC50 = 8.1 nM T52522 CF6X0Z 54580133 EC50 = 173 nM T52522 CN03FM 54582151 EC50 = 5.7 nM T52522 CA74TP 54583092 EC50 = 15 nM T52522 C50PTV 54583100 EC50 = 13 nM T52522 CJC2E3 54586985 EC50 = 10 nM T52522 C2ZYD7 54586986 EC50 = 116 nM T52522 C2IJF0 54591014 EC50 = 0.2512 nM T52522 CWYX94 54757772 EC50 = 14 nM T52522 CRGV73 56597179 EC50 = 10000 nM T52522 CB8O9W 56598831 EC50 = 10000 nM T52522 CQKF90 56598832 EC50 = 10000 nM T52522 CR6PU5 56598833 EC50 = 10000 nM T52522 CRO1Y2 56598967 EC50 = 10000 nM T52522 C43AZK 56658246 EC50 = 0.7943 nM T52522 CCAE43 56658405 EC50 = 0.5012 nM T52522 CMWZ90 56658407 EC50 = 0.5012 nM T52522 CN65GJ 56659408 EC50 = 7.943 nM T52522 CU2C6F 56663238 EC50 = 0.1995 nM T52522 CR29QK 56663519 EC50 = 16.6 nM T52522 CPE84D 56665368 EC50 = 1 nM T52522 C07AEN 56666341 EC50 = 7.943 nM T52522 CEU7B9 56668796 EC50 = 0.3162 nM T52522 C0CS2Z 56670092 EC50 = 2.512 nM T52522 C7D6LT 56670158 EC50 = 5.012 nM T52522 C9CRA4 56672269 EC50 = 0.631 nM T52522 CM3YO8 56672271 EC50 = 0.2512 nM T52522 CO0J8H 56673241 EC50 = 1 nM T52522 CXC4G1 56673609 EC50 = 0.7943 nM T52522 CRSF93 56673674 EC50 = 0.631 nM T52522 CLB1V0 56675663 EC50 = 1 nM T52522 CQO4J2 56677231 EC50 = 4 nM T52522 CE5DQ6 56678849 EC50 = 0.7943 nM T52522 CT2E1Z 56678973 EC50 = 1 nM T52522 CV0L8D 56679937 EC50 > 1000 nM T52522 CDJ2N8 56683262 EC50 = 7.943 nM T52522 C6T7YR 56943485 EC50 = 0.3162 nM T52522 C7DEO8 56943515 EC50 = 0.2512 nM T52522 CZF4B5 56943517 EC50 = 0.631 nM T52522 CJ81YS 56943518 EC50 = 0.1585 nM T52522 C5M0CT 56943545 EC50 = 0.1259 nM T52522 CMUQ15 56943546 EC50 = 0.1585 nM T52522 C1TC7Q 56963799 Ki > 10000 nM T52522 C6YNX5 57391344 EC50 = 1.995 nM T52522 C5YI8R 57391345 EC50 = 6.31 nM T52522 C24QMT 57391346 EC50 = 7.943 nM T52522 CWLO06 57391347 EC50 = 2.512 nM T52522 CL05TF 57391348 EC50 = 39.81 nM T52522 CMZ01K 57391349 EC50 = 50.12 nM T52522 C53OMP 57391554 EC50 = 1 nM T52522 CUV85W 57391792 EC50 = 158.49 nM T52522 C9OE0Q 57393116 EC50 = 50.12 nM T52522 C9EHS4 57393349 IC50 = 0.7943 nM T52522 C68ELZ 57393350 IC50 = 31.62 nM T52522 C1ZTX4 57393524 EC50 = 316.23 nM T52522 CR1XL8 57394848 EC50 = 5.012 nM T52522 CYZD14 57395043 EC50 = 31.62 nM T52522 CKOT20 57395240 EC50 = 79.43 nM T52522 CJI37L 57395241 IC50 = 100 nM T52522 C0B4NR 57396600 IC50 = 251188.64 nM T52522 C3W1UO 57396615 EC50 = 1.995 nM T52522 CX0E5P 57396616 EC50 = 63.1 nM T52522 CVRS85 57397010 EC50 = 100 nM T52522 CR08DF 57398384 EC50 = 0.1259 nM T52522 C2CEB9 57398562 EC50 = 0.3981 nM T52522 C64RIP 57398768 EC50 = 3.981 nM T52522 CPIC27 57398769 IC50 = 199.53 nM T52522 CR1H2F 57400044 IC50 = 100000 nM T52522 C3ZB7F 57400045 EC50 = 1.585 nM T52522 C93GBC 57400228 EC50 = 39.81 nM T52522 C1NGZ7 57400229 EC50 = 2.512 nM T52522 CPJ5T4 57400446 IC50 = 0.631 nM T52522 C3TYE1 57401435 EC50 = 2.512 nM T52522 CM7EN2 57401436 EC50 = 7.943 nM T52522 CPIR67 57402061 IC50 = 15.85 nM T52522 C26XJD 57402248 IC50 = 31.62 nM T52522 C47DOC 57403553 IC50 = 10000 nM T52522 CX49RT 57403562 EC50 = 0.3162 nM T52522 C6YS4T 57403563 EC50 = 39.81 nM T52522 CQAI80 57403815 IC50 = 1.995 nM T52522 CNYB81 59119410 EC50 = 2.512 nM T52522 CW09LS 59119417 EC50 = 7.943 nM T52522 CB47FI 59119455 EC50 = 10 nM T52522 CI3VH0 59119466 EC50 = 6.31 nM T52522 CI9P1B 59119467 EC50 = 2.512 nM T52522 C4UF6I 59119472 EC50 = 7.943 nM T52522 C45JFO 59145957 EC50 = 21 nM T52522 C3WS7G 59707188 EC50 = 23 nM T52522 CGO41Y 59707195 EC50 = 26 nM T52522 C5BSH0 66653268 EC50 = 10000 nM T52522 CS2K0M 66796015 EC50 = 0.1 nM T52522 C3ARI1 67972106 IC50 = 5600 nM T52522 CXJ68U 67972107 IC50 > 20000 nM T52522 CB05ID 67972431 IC50 > 20000 nM T52522 CMG51Y 68807656 Ki = 3.2 nM T52522 CPX1H7 69119729 EC50 = 1 nM T52522 CV57BY 69119831 EC50 = 0.5012 nM T52522 C86CXO 69119890 EC50 = 1.585 nM T52522 C4H3LN 69120058 EC50 = 31.62 nM T52522 CNVH59 69442961 EC50 = 7.943 nM T52522 CKWP40 69447283 EC50 = 39.81 nM T52522 C8DS7F 70684522 EC50 = 138 nM T52522 CONA38 70684846 Ki = 45 nM T52522 CTZ8J0 70686652 EC50 = 165.96 nM T52522 C02NQY 70691181 Ki = 19.4 nM T52522 CBDL19 70792359 IC50 > 20000 nM T52522 C4TWS5 71452172 Ki > 10000 nM T52522 C8U1RC 71558565 EC50 = 0.2512 nM T52522 CG0HF7 73056754 EC50 = 1.63 nM T52522 CE0J8X 73056755 EC50 = 26200 nM T52522 C9HP0N 73056756 Ki = 250 nM T52522 CP9L3Y 73056757 EC50 = 10.19 nM T52522 C9M8NT 73056758 EC50 = 1010 nM T52522 CF6BH0 73056759 Ki = 3419.79 nM T52522 C3K6DW 73057082 Ki = 4740 nM T52522 CNQ7S8 73057083 EC50 = 210 nM T52522 CC65OA 73213195 Ki > 10000 nM T52522 CW83DK 73213196 Ki > 10000 nM T52522 C7TM8S 73349644 EC50 = 50 nM T52522 C74QNU 73352659 EC50 = 40 nM T52522 CG0Z2D 73357212 EC50 = 30 nM T52522 C2E7QW 75201901 Ki = 9300 nM T52522 CVY13Q 76314766 IC50 > 20000 nM T52522 C5ZDK4 76315637 EC50 = 58 nM T52522 CFZU52 76315638 EC50 = 13 nM T52522 C0X7CQ 76315639 EC50 = 120 nM T52522 CGZ5C4 76315640 EC50 = 32 nM T52522 C67YUD 76318362 IC50 > 20000 nM T52522 C1M4TQ 76318363 IC50 > 20000 nM T52522 CCUG71 76318364 IC50 > 20000 nM T52522 C9PM0U 76319327 EC50 = 19 nM T52522 CR05PL 76322043 IC50 > 20000 nM T52522 CQ3CW1 76322044 IC50 > 20000 nM T52522 CFU26T 76322045 IC50 = 2513 nM T52522 CTD25H 76322046 IC50 > 20000 nM T52522 C61AMT 76322047 IC50 > 20000 nM T52522 CI8XA7 76322965 EC50 = 53 nM T52522 CQI0H5 76325667 IC50 > 20000 nM T52522 C6R4BP 76325668 IC50 > 20000 nM T52522 CB71EI 76325669 IC50 > 20000 nM T52522 C03YTR 76329059 EC50 = 19.95 nM T52522 CRW8C5 76329232 IC50 > 20000 nM T52522 C5SKR4 76332892 IC50 = 2471 nM T52522 CMR86G 76332893 IC50 > 20000 nM T52522 CTVI40 76332894 IC50 > 20000 nM T52522 CL7TN0 76332895 IC50 > 20000 nM T52522 C8PGV1 76333795 EC50 = 26 nM T52522 CQ47BW 76336499 IC50 > 20000 nM T52522 C92WBQ 76336500 IC50 > 20000 nM T52522 C8KBZ1 76336501 IC50 = 8451 nM T52522 CQM69X 76336502 IC50 > 20000 nM T52522 CRH70L 87142783 EC50 = 50.12 nM T52522 CZM89H 90644139 EC50 = 2.512 nM T52522 C0N3TA 90644140 EC50 = 199.53 nM T52522 CP14DT 90644141 EC50 = 31.62 nM T52522 C93QFA 90644142 EC50 = 25.12 nM T52522 CE48KB 90644143 EC50 = 1584.89 nM T52522 CW95JO 90644144 EC50 = 158.49 nM T52522 C3T1UD 90644145 EC50 = 398.11 nM T52522 CN8SF5 90644146 EC50 = 501.19 nM T52522 CB7I0W 90644147 EC50 = 1584.89 nM T52522 CZ60EK 90644148 EC50 = 1258.93 nM T52522 CEZ23R 90644149 EC50 = 199.53 nM T52522 C9DTM6 90644150 EC50 = 630.96 nM T52522 C4T1VR 90644151 Ki > 10000 nM T52522 C37DWQ 90644152 EC50 = 1000 nM T52522 C57JOK 90644153 EC50 = 19.95 nM T52522 C6C2HF 90644154 EC50 = 199.53 nM T52522 CNXH73 90645344 EC50 = 0.1259 nM T52522 C9W1FB 90645345 EC50 = 0.5012 nM T52522 CR7OT8 90645346 EC50 = 0.5012 nM T52522 C9A5KY 90645347 EC50 = 0.0631 nM T52522 C1HGJ7 90655864 EC50 = 316.23 nM T52522 CS2JO0 90655865 EC50 = 15.85 nM T52522 CRZL94 90655866 EC50 = 5.012 nM T52522 C53GSE 90655867 EC50 = 10 nM T52522 CEY3D8 90655868 EC50 = 7.943 nM T52522 C25OTU 90655869 EC50 = 12.59 nM T52522 C5UF4C 90666101 EC50 = 74 nM T52522 CDI39M 90666102 EC50 = 26 nM T52522 CU2FI1 90666103 EC50 = 129 nM T52522 C18GXP 90666104 EC50 = 90 nM T52522 C30FIA 90666108 EC50 = 102 nM T52522 CV61GN 90666109 EC50 = 65 nM T52522 C0SIZ8 90666110 EC50 = 22 nM T52522 CZ8I0G 90666112 EC50 = 14 nM T52522 C6LB4R 90666113 EC50 = 36 nM T52522 C5MCU0 90666114 EC50 = 57 nM T52522 C0ZCW5 90666115 EC50 = 20 nM T52522 CC5I0L 90666116 EC50 = 21 nM T52522 CIZ46C 90666117 EC50 = 195 nM T52522 C7WR2F 90666118 EC50 = 24 nM T52522 C6KU1V 90666119 EC50 = 17 nM T52522 CK68NB 90666120 EC50 = 42 nM T52522 CEV61D 90666121 EC50 = 23 nM T52522 CV52KY 90666123 EC50 = 13 nM T52522 CJ5X4F 93382180 Ki = 9 nM T52522 COA3U6 102262219 Ki = 0.48 nM T52522 CZSB43 118710935 Ki = 0.8 nM T52522 CX6NP5 118710936 Ki = 0.6 nM T52522 CB5VH9 118710937 Ki = 2 nM T52522 CDJZ51 118710938 Ki = 97 nM T52522 CQ5Z8V 118710939 Ki = 4.2 nM T52522 CWGD39 118710940 Ki = 0.4 nM T52522 CL8SA7 118710941 Ki = 5.5 nM T52522 CEY68Q 118710942 Ki = 7.1 nM T52522 CM8P2H 118710943 Ki = 15 nM T52522 CHL2U8 118710944 Ki = 149 nM T52522 CVHK79 118710945 Ki = 12 nM T52522 CU68XQ 118710946 Ki = 266 nM T52522 CG8PJ0 118710947 Ki = 6.8 nM T52522 C3GW0U 118710948 Ki = 1.4 nM T52522 C9QB7F 118710949 Ki = 3.9 nM T52522 CMJ0S5 118710950 Ki = 1.7 nM T52522 C6I2UZ 118710951 Ki = 32 nM T52522 CUV5Y0 118715454 EC50 > 30000 nM T52522 CQNL51 118725301 EC50 = 60.26 nM T52522 CTY76J 118737348 EC50 = 0.2512 nM T52522 C6IMH9 118737349 EC50 = 0.3981 nM T52522 CPG45H 118737350 EC50 = 0.1995 nM T52522 CUE90B 118737351 EC50 = 0.2512 nM T52522 C1DZ2G 118737352 EC50 = 0.3162 nM T52522 C5VXT3 118737353 EC50 = 1.585 nM T52522 CP37MC 118737354 EC50 = 0.1585 nM T52522 CGZX73 118737355 EC50 = 0.2512 nM T52522 CB8J7S 118737356 EC50 = 0.7943 nM T52522 CF1HQ8 118737357 EC50 = 3.981 nM T52522 CRE4M1 118737358 EC50 = 0.1 nM T52522 CUN9G8 118737359 EC50 = 1.259 nM T52522 CP6WF1 118737360 EC50 = 0.7943 nM T52522 C1FB4S 122194235 EC50 = 3.7 nM T52522 CDM07Q 122680878 EC50 = 316.23 nM T52522 C4D9QY 127026491 IC50 > 20000 nM T52522 C8MC1I 127028408 Ki = 807 nM T52522 CZ61LK 127034966 IC50 = 501.19 nM T52522 CA0SN5 127034967 IC50 = 100 nM T52522 C7L1DB 127037832 IC50 > 20000 nM T52522 CG84RM 127041558 IC50 = 11000 nM T52522 CS20QX 127041559 IC50 > 20000 nM T52522 CN2T3I 127041869 IC50 = 13400 nM T52522 C2BE3M 127041870 IC50 > 20000 nM T52522 C31SDE 127042181 IC50 > 20000 nM T52522 C35GAL 127045853 Ki = 0.25 nM T52522 C17LBT 127045854 Ki = 13 nM T52522 CJ8GS7 127045855 EC50 = 63.1 nM T52522 C2E1ZA 127046948 Ki = 23 nM T52522 CTI5Z8 127046949 Ki = 6.3 nM T52522 C4D6BQ 127046950 Ki = 18 nM T52522 CM4CQ7 127046951 Ki = 47 nM T52522 C29ERQ 127046952 Ki = 53 nM T52522 C78IFA 127047221 Ki = 850 nM T52522 CZL0U7 127047859 Ki = 2.8 nM T52522 CZ6XL5 127047996 Ki = 610 nM T52522 C50GOC 130442480 Ki > 10000 nM T52522 CM04RF 130442572 Ki = 8600 nM T52522 CAVB41 132584404 Ki > 10000 nM T52522 CBU81N 134149168 Ki > 10000 nM T52522 C1GY2T 135156251 EC50 > 10000 nM T52522 C2QCA5 137631487 IC50 > 20000 nM T52522 C8HPN4 137634334 IC50 > 20000 nM T52522 CZ4TA9 137640201 Ki = 9549.93 nM T52522 C70XZQ 137643636 IC50 > 20000 nM T52522 CL06NY 137648464 IC50 > 20000 nM T52522 CUFO39 137649223 IC50 > 20000 nM T52522 C65XKJ 137653127 IC50 > 20000 nM T52522 C3LG7W 137655838 IC50 > 20000 nM T52522 CN2UE9 137656598 IC50 > 20000 nM T52522 CS8X0I 137660459 Ki = 9 nM T52522 C9C8LN 141465526 EC50 = 50.12 nM T52522 CT9UM2 141465530 EC50 = 316.23 nM T52522 C16DMF 141486999 EC50 = 5100 nM T52522 CP6AM5 145949377 Ki > 100000 nM T52522 CROP78 145949554 Ki > 100000 nM T52522 C8XAH1 145950880 Ki > 100000 nM T52522 C53EGH 145950894 Ki > 100000 nM T52522 C87JIM 145951255 Ki = 31622.78 nM T52522 CQC79A 145951865 Ki > 100000 nM T52522 CUJ2G6 145952345 Ki > 100000 nM T52522 C0UBV8 145955012 Ki > 100000 nM T52522 CMGN62 145956070 Ki = 28183.83 nM T52522 CS93JU 145956073 Ki > 100000 nM T52522 CHXP91 145956144 Ki > 100000 nM T52522 CZK0L8 145956164 Ki > 100000 nM T52522 CRUI17 145956819 Ki = 30199.52 nM T52522 C6I1XE 145956976 Ki = 5011.87 nM T52522 CQO8H5 145958250 Ki > 100000 nM T52522 CC32ZJ 145958632 Ki > 100000 nM T52522 C29YFS 145959974 Ki = 39810.72 nM T52522 C9MSK2 145960116 Ki > 100000 nM T52522 CKE97S 145964215 Ki > 1000000 nM T52522 C24BEA 145965875 Ki = 10400 nM T52522 C07QDS 145966568 Ki = 80400 nM T52522 C8C4YV 145972154 Ki = 4390 nM T52522 CCX0G8 145974110 Ki = 520 nM T52522 CO1SQ3 145977755 Ki = 95400 nM T52522 C18LBV 145978746 Ki = 52300 nM T52522 C72IAC 145980824 EC50 = 5.012 nM T52522 C8EHD9 145981007 EC50 = 10 nM T52522 C4U3RO 145981079 EC50 = 39.81 nM T52522 CU2LP6 145981405 EC50 = 1.995 nM T52522 CG28KC 145981443 IC50 = 210 nM T52522 CB2S3N 145982386 EC50 = 79.43 nM T52522 CBNQ70 145982607 EC50 = 280.8 nM T52522 C6MWR1 145982668 EC50 = 294.5 nM T52522 CFBS76 145983266 EC50 = 8433 nM T52522 CZ60KX 145983355 EC50 = 954.3 nM T52522 COZ4J2 145983711 EC50 = 9842 nM T52522 C9DX1E 145984042 EC50 = 15930 nM T52522 CT4BM0 145984324 EC50 = 1419 nM T52522 CZEM40 145984404 IC50 > 10000 nM T52522 CE5PC2 145984584 EC50 = 52.21 nM T52522 C82AHK 145984792 EC50 = 6058 nM T52522 CFJ6H7 145985170 EC50 = 316.23 nM T52522 CH7MX0 145985242 EC50 = 83.14 nM T52522 C1ZWI5 145986105 EC50 = 117.8 nM T52522 CMD7U6 145986860 IC50 = 20 nM T52522 CD62SW 145987168 EC50 = 1.995 nM T52522 C74LVN 145987415 EC50 = 2.512 nM T52522 CB1T9H 145987609 EC50 = 794.33 nM T52522 CLCV71 145987938 EC50 = 19.95 nM T52522 CK1C0A 145989075 EC50 = 1.585 nM T52522 C0CTI5 145989107 EC50 = 251.19 nM T52522 CA0HG3 145989180 EC50 = 50.12 nM T52522 CUL5A6 145989945 EC50 = 1.26 nM T52522 CO31ZW 145990515 EC50 = 328 nM T52522 C4GV8Q 145990586 IC50 = 1.4 nM T52522 C5F7YS 145990793 EC50 = 3.981 nM T52522 C1J9AT 145991502 EC50 = 630.96 nM T52522 C0SH3Y 145991661 EC50 = 3.162 nM T52522 CAEF85 145992059 EC50 = 630.96 nM T52522 CT6SD4 145992462 EC50 = 12.59 nM T52522 C06QWE 145992510 EC50 = 5.012 nM T52522 CJ8G0D 145992971 EC50 = 50.12 nM T52522 CV7U8T 145994130 EC50 = 10 nM T52522 CC2G1V 146025727 Ki = 5900 nM T52522 C7HM0B 146025801 Ki = 3.3 nM T52522 CKAW68 146025802 Ki = 21 nM T52522 CEP41C 146025803 Ki = 7.2 nM T52522 C6P3SR 153287553 Ki > 10000 nM T52522 CV9G7Z 153287572 Ki > 10000 nM T52522 CO85KL 153287574 Ki > 10000 nM T52522 CB1F6M 155510718 Ki = 1.514 nM T52522 CMJ5H9 155511898 Ki = 26 nM T52522 CKW26I 155512746 Ki = 51 nM T52522 C8P3KR 155512924 Ki = 700 nM T52522 CQ8O2V 155513474 EC50 = 0.08128 nM T52522 CQFN38 155513731 Ki = 420 nM T52522 CRP43D 155514341 Ki = 512 nM T52522 CQP6N7 155515551 Ki = 1.148 nM T52522 C1N6LR 155515718 EC50 = 0.5012 nM T52522 CP0R2N 155515823 IC50 = 6.31 nM T52522 CUM2N4 155515982 Ki = 1800 nM T52522 COD1V4 155516656 Ki = 2000 nM T52522 CERN85 155517986 EC50 = 0.02089 nM T52522 C8NG9I 155518547 Ki = 1.175 nM T52522 CUSA24 155519891 Ki = 575.44 nM T52522 CI9C8O 155521165 Ki = 2200 nM T52522 CI5Z4A 155521390 IC50 = 3.311 nM T52522 CR9DE2 155521528 Ki = 170 nM T52522 CG2F9X 155521599 Ki = 26 nM T52522 CQL75N 155524038 EC50 = 0.1318 nM T52522 C4NOD0 155524193 Ki = 78.6 nM T52522 CWG8V9 155524756 Ki = 1300 nM T52522 CYE26M 155525244 Ki = 0.073 nM T52522 CPCK60 155526570 Ki = 2.9 nM T52522 C5D9JC 155526662 Ki = 740 nM T52522 C46NXV 155527302 Ki = 15 nM T52522 CAQD37 155527582 Ki = 3800 nM T52522 CM78EJ 155527605 IC50 = 8.318 nM T52522 CDJ8F2 155527926 EC50 = 0.2239 nM T52522 CN7D8W 155528927 Ki = 0.8913 nM T52522 CIO7M9 155529446 Ki = 3.4 nM T52522 CUP63K 155529870 Ki = 1.1 nM T52522 CSCN63 155530901 IC50 < 1 nM T52522 CABK31 155530927 IC50 = 1.738 nM T52522 C6K5WZ 155531077 EC50 = 0.2512 nM T52522 CLZY37 155531982 Ki = 3.7 nM T52522 CN90CA 155532901 IC50 = 85.11 nM T52522 CAIC19 155533625 EC50 = 0.04074 nM T52522 CM0EJ2 155534529 Ki = 120 nM T52522 CV23QL 155535986 IC50 = 11.22 nM T52522 CB79ZW 155536080 Ki = 5011.87 nM T52522 CQ70ZB 155536173 EC50 = 0.2188 nM T52522 C0C1ZH 155536314 EC50 = 0.036 nM T52522 C2GLP7 155536373 Ki = 0.955 nM T52522 C30WYL 155536406 Ki = 320 nM T52522 CV7X4Y 155536813 EC50 = 0.04266 nM T52522 CQY6O9 155537285 IC50 = 213.8 nM T52522 CQ0WD1 155537995 Ki = 16.4 nM T52522 C9U1EQ 155539613 Ki = 0.4365 nM T52522 CYH04N 155539979 IC50 = 5.888 nM T52522 C0DQR2 155540000 Ki = 7900 nM T52522 CEX14L 155540608 EC50 = 2.512 nM T52522 CC3FS2 155541417 Ki = 5200 nM T52522 C1U8JI 155541614 EC50 = 0.9333 nM T52522 CYP6C0 155543195 Ki = 920 nM T52522 CZ5F4E 155543358 EC50 = 0.04898 nM T52522 C62AZC 155543518 EC50 = 0.302 nM T52522 CQK0S7 155544582 Ki = 0.7943 nM T52522 CD39HU 155545397 IC50 = 500 nM T52522 C0KO4S 155545790 IC50 = 12.02 nM T52522 CQ29LI 155546387 IC50 = 3.89 nM T52522 CAJ01M 155548071 EC50 = 0.07413 nM T52522 C2SD5W 155548437 Ki = 0.16 nM T52522 C38LYF 155548668 EC50 = 0.07586 nM T52522 C17YQR 155550544 EC50 = 9.12 nM T52522 C65JRG 155550964 EC50 = 0.1514 nM T52522 CA3ST2 155551006 EC50 = 0.5012 nM T52522 C7DE8Z 155551133 EC50 = 0.1622 nM T52522 C3JEN6 155552089 Ki = 3.2 nM T52522 CX8JA1 155552185 Ki = 4500 nM T52522 CUXK56 155552760 IC50 = 83.4 nM T52522 C28YNT 155555687 Ki = 57 nM T52522 CTPM05 155557081 IC50 = 213.8 nM T52522 CB85MA 155557083 EC50 = 0.05012 nM T52522 CF8R5C 155558987 Ki = 6900 nM T52522 CD1S5X 155559932 IC50 = 14.13 nM T52522 C7EVF6 155559960 Ki = 0.3802 nM T52522 C04UEW 155561031 Ki = 20 nM T52522 CKM05W 155563970 IC50 = 2.188 nM T52522 CR8W7Y 155564079 EC50 = 0.06457 nM T52522 C8C0RW 155564274 Ki = 1400 nM T52522 CL43AX 155564340 EC50 = 0.05129 nM T52522 CD78XW 155564766 EC50 = 0.04074 nM T52522 CS0U7F 155564992 IC50 = 64.57 nM T52522 CZ51GL 155565922 IC50 = 6.457 nM T52522 C5KDA9 155566405 Ki = 10.3 nM T52522 CA05IO 155567283 EC50 = 0.07413 nM T52522 CUT84A 155568798 EC50 > 100000 nM T52522 C9S1RP 155568878 IC50 = 13.8 nM T52522 CMU1C9 155569481 Ki = 0.7586 nM T52522 CP9TR0 10324985 Ki = 60.6 nM T52522 CF40LD 44349237 IC50 = 220 nM T52522 CTNO31 44349323 IC50 = 2400 nM T52522 C91AXH 44349356 IC50 = 370 nM T52522 C9JZ7V 44349357 IC50 = 3400 nM T52522 C5TWZ0 44349367 IC50 = 5600 nM T52522 CE2XL3 44349378 IC50 = 1200 nM T52522 C5ELB7 44349379 IC50 = 1200 nM T52522 D01JXM 46222048 Ki > 1000 nM T52522 D01OIK 155774 EC50 = 707.95 nM T52522 D01WWC 16573 Ki > 950 nM T52522 D02DKX 5311116 EC50 = 10000 nM T52522 D02QPP 688467 EC50 = 4.7 nM T52522 D02VPW 6603756 Ki = 0.1 nM T52522 D03DET 10287730 Ki = 1995.26 nM T52522 D03VHK 10028830 EC50 = 23490 nM T52522 D04BYL 10352428 Ki = 70100 nM T52522 D04HXF 4080436 Ki = 1.2 nM T52522 D04JGC 688468 EC50 = 0.3 nM T52522 D05GDP 599482 Ki > 10000 nM T52522 D05JKG 68770 Ki = 900 nM T52522 D05RWZ 6603724 Ki = 15800 nM T52522 D05ZUX 44207909 Ki >= 1000 nM T52522 D09PIN 3378093 Ki > 1000 nM T52522 D09RPR 16737207 Ki > 10000 nM T52522 D0A0KP 37990 EC50 = 0.054 nM T52522 D0A4FU 2769774 Ki = 7 nM T52522 D0A9ED 71739 Ki = 0.03 nM T52522 D0C6CZ 23968266 Ki = 0.145 nM T52522 D0H2WQ 54562 Ki = 100000 nM T52522 D0L5MW 181743 Ki > 10000 nM T52522 D0OL3X 667688 EC50 = 8.5 nM T52522 D0R3GW 10296414 Ki < 501.19 nM T52522 D0T2RY 9948320 Ki >= 1000 nM T93653 D0V3YT 10324367 IC50 = 75 nM T93653 D0X9CH 3010818 IC50 = 1350 nM T93653 D0J6AU 10152654 IC50 = 762 nM T93653 D0T5PH 6918602 Ki = 0.063 nM T93653 CIF9A2 95706 IC50 = 7200 nM T93653 C5YNV4 161091 IC50 = 4700 nM T93653 C4U5MD 202918 IC50 > 50000 nM T93653 C62DWI 231061 IC50 = 10000 nM T93653 C31BIK 832505 IC50 = 5000 nM T93653 C9RQ2F 2848907 IC50 = 2000 nM T93653 CR2ND4 5287468 Ki = 1.8 nM T93653 CW6D7Z 5287498 IC50 = 7100 nM T93653 CWOL57 5339865 IC50 = 15000 nM T93653 CV5UC4 5378702 IC50 = 48000 nM T93653 CWK27I 5487772 Ki = 1000 nM T93653 C0XQP7 6917747 IC50 > 100000 nM T93653 CN26IL 9547980 Ki > 30000 nM T93653 CF9N8S 9798626 IC50 = 44000 nM T93653 CNU47F 9834637 IC50 = 20000 nM T93653 C4QGU3 9998312 Ki = 1100 nM T93653 CJQE31 10016895 Ki = 4200 nM T93653 CLB5G0 10025017 IC50 = 79 nM T93653 C1QB5U 10063343 IC50 = 9900 nM T93653 CFC3Q8 10120133 IC50 = 34000 nM T93653 C6AZ3B 10120903 IC50 = 36000 nM T93653 CDX7R4 10164961 IC50 = 5600 nM T93653 C5B1HM 10165557 IC50 = 1600 nM T93653 CTJ7R3 10166544 IC50 = 430 nM T93653 C4M3SG 10186046 IC50 = 230000 nM T93653 C0SF7U 10187920 IC50 = 130 nM T93653 CS3IP7 10210867 IC50 = 5000 nM T93653 CT8K5D 10231379 IC50 = 170 nM T93653 C4OZ5K 10231447 IC50 = 1200 nM T93653 CV9LB1 10302710 IC50 = 2800 nM T93653 CUQ2R3 10303526 IC50 = 4500 nM T93653 CV5S7B 10303657 IC50 = 36000 nM T93653 C54TDE 10385901 Ki = 1200 nM T93653 C7BI2T 11009218 IC50 = 4700 nM T93653 CFI8L5 11502586 IC50 = 29 nM T93653 CFVX76 11580650 Ki = 10000 nM T93653 CILB73 11649751 Ki > 20000 nM T93653 C3JO1P 12262704 IC50 > 50000 nM T93653 C31MCN 13186896 IC50 > 100000 nM T93653 C6XPN4 16664855 IC50 = 131 nM T93653 CP1A6L 20262575 IC50 = 2100 nM T93653 CQU38W 24900755 IC50 = 3317 nM T93653 C2S8VB 24901099 IC50 = 158 nM T93653 CIN28B 24901100 IC50 = 1289 nM T93653 CD2EH0 24901101 IC50 = 894 nM T93653 CS7B3F 24901102 IC50 > 10000 nM T93653 CC7TV3 25204336 IC50 > 10000 nM T93653 C73KLE 25209862 IC50 = 140 nM T93653 CZS24P 42633520 IC50 = 79 nM T93653 CI78XT 42633521 IC50 = 69 nM T93653 CZ6B1F 42635119 IC50 = 28 nM T93653 C25ELB 44143088 IC50 = 239.88 nM T93653 C9QDC0 44143091 IC50 = 70794.58 nM T93653 CJA68L 44224113 IC50 = 794.33 nM T93653 C2V5ZT 44224114 IC50 = 6309.57 nM T93653 C0U9VJ 44224115 IC50 = 398.11 nM T93653 C0MZ9D 44224116 IC50 = 6309.57 nM T93653 CEJ82A 44224117 IC50 = 1000 nM T93653 C0KL7D 44224118 IC50 = 794.33 nM T93653 CE9S0M 44224119 IC50 = 5011.87 nM T93653 CV1W0Z 44224120 IC50 = 199.53 nM T93653 C5LDK7 44224121 IC50 = 1584.89 nM T93653 C8UF5Q 44224122 IC50 = 3981.07 nM T93653 C9YHC5 44224123 IC50 = 199.53 nM T93653 CA26RI 44224124 IC50 = 3981.07 nM T93653 CU0PI2 44224125 IC50 > 10000 nM T93653 CRL79W 44224126 IC50 = 3162.28 nM T93653 C3T0QO 44224127 IC50 = 1000 nM T93653 C81EVM 44224128 IC50 = 1258.93 nM T93653 C7IY8P 44224129 IC50 = 1258.93 nM T93653 CYG02V 44224130 IC50 = 2511.89 nM T93653 CJS1B9 44224131 IC50 = 251.19 nM T93653 CN5O8S 44224132 IC50 = 501.19 nM T93653 C2Q3RP 44224133 IC50 = 501.19 nM T93653 CZX62T 44224134 IC50 = 501.19 nM T93653 CP3YA9 44224135 IC50 = 199.53 nM T93653 CSZH31 44224136 IC50 = 398.11 nM T93653 C2J6MW 44397423 IC50 = 1300 nM T93653 CRSF50 44397609 IC50 = 1700 nM T93653 CHWX97 44397693 IC50 = 14000 nM T93653 CD18YP 44402055 IC50 = 340 nM T93653 CU8TB9 44402056 IC50 = 390 nM T93653 CD4TP7 44402158 IC50 = 290 nM T93653 CO6BG2 44402160 IC50 = 180 nM T93653 C0AJC4 44402175 IC50 = 2000 nM T93653 CX9O2Q 44402263 IC50 = 2800 nM T93653 C89MOT 44402291 IC50 = 190 nM T93653 CS6X7V 44426055 IC50 = 5166 nM T93653 C8IB2W 44426056 IC50 > 100000 nM T93653 C8Z4WO 44459967 IC50 = 831.76 nM T93653 C86ORE 44459987 IC50 = 181.97 nM T93653 C4YAJ7 46228924 IC50 > 10000 nM T93653 CC2N0F 46842579 IC50 > 10000 nM T93653 CV6SW4 46842581 IC50 > 10000 nM T93653 CM2D1G 46842582 IC50 > 10000 nM T93653 CIU1R5 46842626 IC50 > 10000 nM T93653 C37OSC 46842709 IC50 > 10000 nM T93653 C37RZT 49862146 IC50 > 10000 nM T93653 CJ0HY8 49862186 IC50 > 10000 nM T93653 CDC64G 52941172 IC50 > 10000 nM T93653 C71VFU 52941469 IC50 = 29.5 nM T93653 CW05MV 52942797 IC50 = 16.6 nM T93653 CQDG96 52943578 IC50 = 1122 nM T93653 C75SHQ 52948860 IC50 = 36.3 nM T93653 CO95XY 53316985 Ki = 500 nM T93653 CH9KW3 53318269 Ki = 1700 nM T93653 CJ3PN0 53319501 IC50 > 10000 nM T93653 C7V2DA 53322116 IC50 > 10000 nM T93653 CQ8O1R 53322117 IC50 > 10000 nM T93653 C19BCV 53326179 Ki = 4400 nM T93653 CBY72G 66572720 Ki = 800 nM T93653 C34GCU 66572722 IC50 = 16000 nM T93653 CHWA75 66572723 IC50 = 15000 nM T93653 C78CAD 66572724 IC50 = 8500 nM T93653 CAF7U2 66572726 Ki = 1300 nM T93653 C3V1BY 66572849 IC50 = 1700 nM T93653 C1Q5WX 66572850 IC50 = 8200 nM T93653 CLJ58E 66572851 Ki = 400 nM T93653 C3VLY0 66572852 IC50 = 18000 nM T93653 C4TXD6 66572853 IC50 = 4900 nM T93653 CZI74Q 70683995 IC50 = 25000 nM T93653 CADN96 70683996 IC50 > 50000 nM T93653 CM5C8Q 70686123 Ki = 1100 nM T93653 CN4QX8 70686124 IC50 = 9000 nM T93653 CBV9F6 70688255 IC50 = 3500 nM T93653 C47WPT 70688256 IC50 = 6900 nM T93653 CMW4T8 70688257 IC50 = 6800 nM T93653 CLE18H 70692439 IC50 = 1500 nM T93653 CAB1L6 70692440 Ki = 800 nM T93653 C5D8SA 70692441 IC50 > 50000 nM T93653 CGV1W9 70696541 IC50 > 50000 nM T93653 CXY0A7 70696542 IC50 = 12300 nM T93653 CAN6X5 71656574 IC50 = 1043 nM T93653 CTZJ19 155513164 IC50 = 420 nM T93653 CYN70B 155529581 IC50 = 700 nM T93653 C6T3XK 155551861 IC50 = 1400 nM T93653 C58OLD 44517711 IC50 = 39.81 nM T93653 CT3S1I 44517712 IC50 = 100 nM T93653 CFT38D 45267632 IC50 = 158.49 nM T93653 COU83P 45267640 IC50 = 25.12 nM T93653 C1U4IF 45267645 IC50 = 3.162 nM T93653 CDG5S8 45268499 IC50 = 1584.89 nM T93653 CV8PZ3 45268510 IC50 > 10000 nM T93653 C89ADF 45269361 IC50 = 1584.89 nM T93653 C58PZI 45269375 IC50 = 158.49 nM T93653 C5O9EF 45270206 IC50 = 6.31 nM T93653 C07ADH 45270207 IC50 = 1.995 nM T93653 CVGE81 45270212 IC50 = 7.943 nM T93653 C78EXG 45271021 IC50 = 3981.07 nM T93653 C5MBC4 45271038 IC50 = 6.31 nM T93653 C65QLD 45271887 IC50 > 7943.28 nM T93653 CIL8O6 45271888 IC50 = 3981.07 nM T93653 CLFD35 45272742 IC50 = 3162.28 nM T93653 C3WF8S 45272748 IC50 > 10000 nM T93653 CQO98K 45272752 IC50 = 63.1 nM T93653 C9A0IH 45272753 IC50 = 19.95 nM T93653 CSYU09 45273681 IC50 = 3162.28 nM T93653 D04URI 19093029 Ki = 200 nM T93653 D0Y5IQ 44255320 IC50 = 10000 nM T14181 C4ZB6V 145949328 Ki = 18400 nM T14181 C7HX2P 145950658 Ki = 461000 nM T14181 CCH9D1 145950714 Ki = 115000 nM T14181 C2UGH9 145951072 Ki = 41400 nM T14181 CX63BS 145951196 Ki = 240 nM T14181 CI46QL 145951895 Ki = 11300 nM T14181 C7BL4X 145951965 Ki = 26800 nM T14181 CLN89R 145952155 Ki = 61200 nM T14181 CL9Y3T 145952242 Ki = 130300 nM T14181 C6WF1I 145952861 Ki > 100000 nM T14181 C53MEX 145953699 Ki = 98000 nM T14181 C02WMA 145954911 Ki = 58200 nM T14181 CD4Q5R 145954958 Ki = 90 nM T14181 C7H8VS 145955044 Ki = 14300 nM T14181 C1J3LZ 145955095 Ki = 3400 nM T14181 C5YQ0B 145955211 Ki = 6100 nM T14181 CZWT76 145955490 Ki = 4700 nM T14181 CYZV20 145955959 Ki = 2200 nM T14181 CCG47F 145956151 Ki = 3200 nM T14181 CGR21E 145956871 Ki = 1400 nM T14181 CQT53G 145957102 Ki = 122600 nM T14181 CY1J9A 145957770 Ki = 210 nM T14181 C52TRH 145958419 Ki = 26300 nM T14181 C6I3LJ 145958437 Ki = 510 nM T14181 C0T7MC 145958949 Ki = 720 nM T14181 CK1IS4 145959136 Ki = 1890 nM T14181 C18PYI 145959769 Ki > 500000 nM T14181 C4B2OD 145959845 Ki = 8500 nM T14181 CF3V1K 145960130 Ki = 43200 nM T14181 CHB89W 145960230 Ki = 380 nM T14181 CO9U7B 145971470 Ki = 11200 nM T14181 C5VEI3 145973349 Ki = 22800 nM T14181 CD13JH 145973367 Ki = 340 nM T04361 D0E3TC 44259 IC50 = 66.2 nM T04361 C9D5CL 9799061 IC50 = 1300 nM T04361 CK2J3G 9863776 IC50 = 5.6 nM T04361 C0UL1D 9863860 IC50 = 2600 nM T04361 CW46YG 9929643 IC50 = 33 nM T04361 C0V7UW 9958506 IC50 > 11000 nM T04361 C5UG6X 10114595 Ki = 1300 nM T04361 C8K9HL 10142476 Ki = 130 nM T04361 CN37YZ 10207985 Ki = 2500 nM T04361 C8BHJ3 10226185 Ki = 800 nM T04361 C78SMB 10227510 Ki = 15 nM T04361 CXN06I 10227557 Ki = 2500 nM T04361 C0SR5Y 10278151 Ki = 30 nM T04361 C9BH5R 10959857 IC50 > 30000 nM T04361 CCEJ71 11406978 IC50 = 380 nM T04361 CU0E8O 11690457 Ki = 2700 nM T04361 CB0AP2 11705863 Ki > 4000 nM T04361 C47NEQ 11728572 IC50 = 990 nM T04361 CM4F0B 21899142 Ki = 700 nM T04361 CLBP72 24798571 IC50 > 10000 nM T04361 C0VIX4 44219633 Ki > 4000 nM T04361 CV17TJ 46888372 IC50 = 10000 nM T04361 CEQN27 52936621 Ki = 860 nM T04361 C79CBU 53377635 IC50 = 9100 nM T04361 C91QFZ 53378283 IC50 = 1100 nM T04361 C7SD4U 53378486 IC50 = 200 nM T04361 C9KU7J 53378487 IC50 = 5200 nM T04361 C6WTM3 53378489 IC50 = 3100 nM T04361 CC75QD 53378696 IC50 = 1800 nM T04361 CX9WJ0 53378698 IC50 = 8000 nM T04361 C0N2OE 53378808 IC50 = 4000 nM T04361 C1T2KG 53378914 IC50 = 44 nM T04361 CD4UT8 53378915 IC50 = 2700 nM T04361 CZSX35 53379038 IC50 = 12 nM T04361 CPR38O 53379040 IC50 = 10 nM T04361 CI70CT 57345538 IC50 = 650 nM T04361 COH62U 60097413 IC50 > 10000 nM T04361 C1MR8Q 60097495 IC50 > 10000 nM T04361 CA7DO0 66759456 IC50 = 1500 nM T04361 CCS0D6 66759463 IC50 = 4400 nM T04361 CBX0G2 66759517 IC50 = 4500 nM T04361 C45DSL 66759520 IC50 = 520 nM T04361 CR05YE 66759532 IC50 = 610 nM T04361 CWA16U 66759542 IC50 = 3100 nM T04361 C6A3TN 66759619 IC50 = 1700 nM T04361 CW4C1V 66759861 IC50 = 370 nM T04361 C5BD1X 66759873 IC50 = 9000 nM T04361 CAL28J 66759967 IC50 = 1200 nM T04361 CF8R0H 66760038 IC50 = 470 nM T04361 CEDB58 66760097 IC50 = 440 nM T04361 CA90UQ 66760159 IC50 = 1900 nM T04361 CZ39PX 66760160 IC50 = 340 nM T04361 C7LOI5 66760328 IC50 = 1800 nM T04361 C0M8JY 66760335 IC50 = 1700 nM T04361 CCE1H2 66760342 IC50 = 510 nM T04361 CP2A7S 66760349 IC50 = 1200 nM T04361 CY36UH 66760355 IC50 = 18 nM T04361 CXU42A 66760411 IC50 = 1000 nM T04361 CF71QO 66760445 IC50 = 110 nM T04361 C0X2TA 66760450 IC50 = 1100 nM T04361 CB0ML5 66760507 IC50 = 500 nM T04361 CIGD24 66760608 IC50 = 1000 nM T04361 C8DL9V 66760658 IC50 > 20000 nM T04361 CE73VM 66760663 IC50 = 1600 nM T04361 CMW54N 66760714 IC50 = 4400 nM T04361 C1S7ZR 66760763 IC50 = 530 nM T04361 CE20FQ 66760840 IC50 = 15 nM T04361 CW7V4C 66760895 IC50 > 10000 nM T04361 CQUF13 66760947 IC50 = 2800 nM T04361 CZ5JA1 66761050 IC50 = 3000 nM T04361 CP94KX 66761096 IC50 = 190 nM T04361 CLQ51N 66761102 IC50 = 1000 nM T04361 CV63UL 67240318 IC50 > 10000 nM T04361 CA7KJ1 68068082 IC50 = 690 nM T04361 COJ81H 68068167 IC50 = 1200 nM T04361 CAJ12E 68810830 IC50 = 50 nM T04361 CEBO91 71452977 IC50 > 10000 nM T04361 CBP84Y 71543324 IC50 = 8 nM T04361 CMLF37 71814652 IC50 = 17 nM T04361 CPNQ29 71814653 IC50 = 130 nM T04361 CY21KG 71814654 IC50 = 43 nM T04361 CJ98FV 71814655 IC50 = 45 nM T04361 C9GS6R 71814656 IC50 = 20 nM T04361 CW7D9Z 73212018 IC50 = 156 nM T04361 C5N1VZ 102581295 IC50 > 10000 nM T04361 C6I9TF 118713989 IC50 > 30000 nM T04361 C9YEZ7 122193348 IC50 > 30000 nM T04361 CAL7H3 122194136 IC50 = 77 nM T04361 CN8LF4 122194137 IC50 = 360 nM T04361 CR6L9A 122194138 IC50 = 2600 nM T04361 C5ABP9 122194139 IC50 = 8900 nM T04361 CM94KB 122194140 IC50 > 30000 nM T04361 C70XOG 122490483 IC50 = 34 nM T04361 C1Z3SF 127048450 IC50 = 260 nM T04361 C61DZB 127048451 IC50 = 1300 nM T04361 CZKA30 127049266 IC50 = 1600 nM T04361 CSD1B0 127052398 IC50 = 20000 nM T04361 C8ARK0 131801160 IC50 = 50 nM T04361 C0AV5D 131801161 IC50 = 7.6 nM T04361 CB3C0Z 132819859 IC50 = 3.3 nM T04361 CK6Z5F 132819860 IC50 = 25 nM T04361 CR3C9O 132819862 IC50 = 5.1 nM T04361 CAG60V 132819865 IC50 = 7.3 nM T04361 CE4Z3X 132819866 IC50 = 7 nM T04361 C8IZB3 134129887 IC50 = 950 nM T04361 C84IXK 134130027 IC50 = 2750 nM T04361 C3TW9Y 134130036 IC50 = 4.6 nM T04361 CTDB31 134130124 IC50 = 3010 nM T04361 CZA37N 134130230 IC50 = 83 nM T04361 C5N0CA 134130303 IC50 = 1.7 nM T04361 C4S7VK 134130361 IC50 = 75 nM T04361 C71ATR 134130387 IC50 = 1640 nM T04361 C2IB7F 134130412 IC50 = 3.2 nM T04361 C57PSE 134130572 IC50 = 1630 nM T04361 CH7A9R 134130612 IC50 = 57 nM T04361 CEH49U 134130924 IC50 = 4.4 nM T04361 CV3W7U 134131236 IC50 = 342 nM T04361 COL93E 134131237 IC50 = 92 nM T04361 CGBZ13 134843302 IC50 = 1000 nM T04361 CG2LO6 135567179 IC50 = 2.3 nM T04361 C3QGA1 135567180 IC50 = 13 nM T04361 CAX7S0 135567181 IC50 = 11 nM T04361 CWL82V 136211071 IC50 = 41 nM T04361 C2DHW3 136211072 IC50 = 6.7 nM T04361 CA8X5T 136211073 IC50 = 5.8 nM T04361 CACV01 136211074 IC50 = 15 nM T04361 C8A6RC 136254416 IC50 = 500 nM T04361 C3MK9W 136807986 IC50 > 10000 nM T04361 CPOE67 137205231 IC50 = 3.5 nM T04361 C8I7RQ 137205232 IC50 = 220 nM T04361 CA53LC 137205233 IC50 = 7.3 nM T04361 CA37ZE 137205234 IC50 = 3 nM T04361 CH8SO0 137205235 IC50 = 5.2 nM T04361 CZD1C0 137205236 IC50 = 5 nM T04361 C73OTH 137205237 IC50 = 9.3 nM T04361 C9GOK2 145961605 IC50 = 1640 nM T04361 CDHY40 145961984 IC50 = 25 nM T04361 C7OT1V 145962571 IC50 = 1230 nM T04361 CP58OY 145963683 IC50 = 33 nM T04361 COZA72 155415442 IC50 = 224 nM T04361 C8UOT3 155415499 IC50 = 543 nM T04361 CMJZ23 155415509 IC50 = 1490 nM T04361 C09YSN 155415512 IC50 = 5460 nM T04361 C59VKN 155415568 IC50 = 1890 nM T04361 C2MD1Q 155513187 IC50 > 10000 nM T04361 C68GMW 155538446 IC50 = 36000 nM T04361 CY6Q8S 155554337 IC50 = 18000 nM T04361 CO2I4P 155559898 IC50 = 1200 nM T04361 C13GYL 127031746 IC50 < 5000 nM T04361 D0J3LR 11634725 Ki = 3000 nM T05409 D0I0EG 44093 IC50 = 830000 nM T05409 D0U2JP 4369359 IC50 > 100000 nM T05409 D09JES 6324648 IC50 = 0.6 nM T05409 D02DLE 132968 IC50 = 0.9 nM T05409 D04LAQ 443380 IC50 = 7.8 nM T05409 D04MBS 9801007 IC50 = 6 nM T05409 D05UQD 656629 IC50 = 0.1995 nM T05409 D06WBA 123742 IC50 = 9.4 nM T05409 D0I5QZ 9998020 IC50 = 400 nM T05409 D0K9YR 9810328 IC50 = 90 nM T05409 D0T2IQ 443600 IC50 = 6700 nM T05409 CU4AG9 122116 IC50 = 65 nM T05409 C15MKE 124786 IC50 = 1.4 nM T05409 CHG65Y 1590669 Ki = 37000 nM T05409 C3UYH5 1590673 Ki = 25000 nM T05409 CSE85T 2828746 IC50 = 20000 nM T05409 C79HSA 2828749 IC50 = 20000 nM T05409 CY36MH 4369380 Ki = 1.5 nM T05409 CC5O4E 4369384 IC50 = 9400 nM T05409 C53BJS 7059511 Ki = 1.7 nM T05409 CQ53EX 9796137 IC50 = 44000 nM T05409 CMIP58 9806479 IC50 = 5 nM T05409 CXN8M1 9822830 IC50 = 48 nM T05409 CRF51I 9839564 IC50 = 0.9 nM T05409 CZ2HC0 9840687 IC50 = 4 nM T05409 C2MEU1 9844054 IC50 = 4 nM T05409 C02WVA 9862743 IC50 = 60 nM T05409 CYV4Z5 9863167 IC50 = 2300 nM T05409 C2S1ZR 9866271 IC50 = 313 nM T05409 C96UPA 9884141 IC50 = 15000 nM T05409 CZ54NX 9925732 IC50 = 2 nM T05409 CVPG59 9932329 IC50 = 10 nM T05409 COH8P4 9949799 IC50 = 18.9 nM T05409 C2EF4O 9951444 IC50 = 96 nM T05409 CI2HX5 9969592 IC50 = 11 nM T05409 CC60TG 9976354 IC50 = 550 nM T05409 C1FM2C 9979153 IC50 = 8600 nM T05409 C5UH9J 10041763 IC50 = 8 nM T05409 CMD3J1 10047309 IC50 = 2.1 nM T05409 C32OGJ 10071569 IC50 = 3 nM T05409 C43WIP 10107035 IC50 = 1.3 nM T05409 C1YM9K 10110899 IC50 = 3.7 nM T05409 C6NDV0 10132004 IC50 = 292 nM T05409 CG0DW7 10141595 IC50 > 100000 nM T05409 CDT6V1 10379000 Ki = 0.7 nM T05409 CWQ16X 10400639 Ki = 162 nM T05409 CEI64K 10426451 IC50 = 14 nM T05409 CX78MU 10432045 IC50 = 9 nM T05409 C8GRN2 10444857 Ki = 4.9 nM T05409 CX38EB 10467565 IC50 > 100000 nM T05409 C4VN0M 10494952 IC50 = 7 nM T05409 C69RND 10496022 IC50 = 4 nM T05409 CTPC82 10501144 IC50 = 6300 nM T05409 COZR84 10505477 IC50 = 2500 nM T05409 C87HBU 10518365 IC50 = 11000 nM T05409 CM1CJ3 10528823 IC50 = 40000 nM T05409 CG0AN8 10601571 IC50 = 5800 nM T05409 C5VGI8 10622593 IC50 = 6700 nM T05409 C7UH9R 10647129 IC50 = 1200 nM T05409 CNJ2K9 10647364 IC50 = 10700 nM T05409 C02PTU 10648112 IC50 = 6200 nM T05409 CW7GR6 10648756 IC50 = 6300 nM T05409 CQN7S4 10664538 IC50 = 67 nM T05409 CI19VE 10669956 IC50 = 10000 nM T05409 CY61XN 10689164 IC50 = 900 nM T05409 CA14CE 10691661 IC50 = 23000 nM T05409 C4Z0CX 10694200 IC50 = 640 nM T05409 C82VZE 10696749 IC50 = 860 nM T05409 C4S3EZ 10710922 IC50 = 8 nM T05409 CSJC70 10715413 IC50 = 55000 nM T05409 CZC4M7 10719503 IC50 = 6500 nM T05409 CI4SQ2 10732349 IC50 > 100000 nM T05409 CAD84L 10735551 IC50 = 27 nM T05409 C6IB1M 10740493 IC50 = 407 nM T05409 CZAO16 10744617 IC50 = 250 nM T05409 CT78AR 10759255 IC50 = 445 nM T05409 C7O6RU 10759256 IC50 = 27 nM T05409 CVA35S 10763731 IC50 = 19000 nM T05409 CGE6W5 10764686 IC50 = 15000 nM T05409 C57SVI 10766810 IC50 = 7000 nM T05409 CX34MD 10768671 IC50 = 730 nM T05409 C1UF0K 10791459 IC50 = 1300 nM T05409 CJP19Q 10829413 IC50 = 26000 nM T05409 CFUE14 10829618 IC50 = 3 nM T05409 C6B4OW 10834551 IC50 = 948 nM T05409 CC0MU7 11192220 IC50 > 100000 nM T05409 CLD37R 11494779 IC50 = 283 nM T05409 C3A9PM 11495237 IC50 > 3000 nM T05409 CIJA12 11515481 IC50 = 1710 nM T05409 C6ZAT5 11515677 IC50 = 3100 nM T05409 CB6LO5 11515875 IC50 = 150 nM T05409 C27CVU 11516039 IC50 = 1500 nM T05409 CNQ9H4 11516163 IC50 = 120 nM T05409 CE34MT 11522221 IC50 = 237 nM T05409 CSIJ47 11531417 IC50 = 195 nM T05409 C1YG8Q 11537626 IC50 = 890 nM T05409 C3PF8I 11544123 IC50 = 377 nM T05409 C81ZNF 11545107 IC50 = 38 nM T05409 CF5H2P 11551902 IC50 = 313 nM T05409 CE3HA6 11556698 Ki = 6700 nM T05409 CH6JG7 11559079 IC50 = 374 nM T05409 C6B5XD 11561143 IC50 = 1139 nM T05409 C91OHX 11566264 IC50 = 213 nM T05409 CTX2W5 11566540 IC50 = 84 nM T05409 CRN1S2 11573732 IC50 > 3000 nM T05409 C5AN1O 11589433 IC50 = 30 nM T05409 C19WSH 11595694 IC50 > 2000 nM T05409 CIJ6B4 11603744 IC50 = 46 nM T05409 CH6ZB0 11610321 IC50 = 124 nM T05409 CU56XA 11631338 IC50 > 2000 nM T05409 CK1OF5 11639199 IC50 > 2000 nM T05409 C95XBL 11645797 IC50 = 700 nM T05409 CFB27N 11646207 IC50 = 184 nM T05409 CZ0I7M 11652422 IC50 = 1500 nM T05409 C3GK4C 11652641 IC50 > 2000 nM T05409 C8E1TB 11652860 IC50 = 530 nM T05409 CZ1LE6 11659857 IC50 = 176 nM T05409 CT61SY 11661034 IC50 = 1060 nM T05409 CCZU50 11661185 IC50 = 96 nM T05409 CO3EB9 11666940 IC50 = 82 nM T05409 C1PRY4 11682031 IC50 = 384 nM T05409 CE1Z3R 11682380 IC50 = 370 nM T05409 C5QXE9 11688419 IC50 = 1710 nM T05409 CWBC32 11689439 IC50 = 297 nM T05409 C10CKM 11704532 IC50 > 10000 nM T05409 C9WK5G 11754555 IC50 = 2070 nM T05409 COT0R7 11792153 IC50 = 82 nM T05409 C09SYT 13178368 IC50 = 15 nM T05409 CHS29Y 14390729 IC50 = 6.6 nM T05409 CLH8D1 15380810 IC50 = 1 nM T05409 CQ20VS 15380813 IC50 = 64 nM T05409 CFX03B 15380816 IC50 = 560 nM T05409 CR40IL 15380817 IC50 = 14 nM T05409 C24BMZ 15380820 IC50 = 0.6 nM T05409 C7R3WN 15380821 IC50 = 3.1 nM T05409 CQGY31 15838528 IC50 = 175 nM T05409 C9TS8Q 15838530 IC50 = 1124 nM T05409 C29DIA 15978653 IC50 = 10.5 nM T05409 CQRX89 18980765 IC50 = 3.5 nM T05409 C80FOI 18980791 IC50 = 2.5 nM T05409 C5PE7J 18980806 IC50 = 3.1 nM T05409 C9X6KQ 18980810 IC50 = 9 nM T05409 CY6KG0 18980812 IC50 = 5.2 nM T05409 C1T2YW 21757876 IC50 = 4 nM T05409 C19LUX 22874513 IC50 > 1000 nM T05409 CL03XM 22874515 IC50 = 83 nM T05409 C3UQD8 22874522 IC50 > 1000 nM T05409 CO1P3U 22874524 IC50 > 1000 nM T05409 C4EY5Q 22874526 IC50 = 940 nM T05409 CGV6A0 22874530 IC50 > 1000 nM T05409 C6FVA5 23285617 IC50 = 2 nM T05409 C2MV9X 24882714 IC50 = 650 nM T05409 C0U8AZ 25015303 IC50 > 50000 nM T05409 CP2LY7 25033280 Ki = 13 nM T05409 C4YKQ1 25033281 Ki = 2.6 nM T05409 C0TR3U 25190005 IC50 = 15.85 nM T05409 C7RS3Y 25195667 IC50 = 30000 nM T05409 C7IHC9 44207184 IC50 = 7000 nM T05409 CR01EW 44256381 IC50 = 7000 nM T05409 C5EMQ6 44264193 IC50 = 6.3 nM T05409 CNG1L3 44266455 IC50 = 0.7 nM T05409 C41APY 44266469 IC50 = 0.6 nM T05409 C49ZRD 44266477 IC50 = 8.8 nM T05409 CGO98H 44266483 IC50 = 1.46 nM T05409 C8R9ES 44266484 IC50 = 0.74 nM T05409 CI3S2Y 44266520 IC50 = 17 nM T05409 C7GOP6 44266525 IC50 = 4.8 nM T05409 CI5M9G 44266561 IC50 = 2.5 nM T05409 CI73GK 44267283 IC50 = 2 nM T05409 COA58H 44267301 IC50 = 2 nM T05409 CWA84R 44267309 IC50 = 16 nM T05409 CS0D9T 44267339 IC50 = 4 nM T05409 C68TCF 44267348 IC50 = 5.9 nM T05409 C7RC8Y 44267350 IC50 = 65 nM T05409 CZGF30 44267353 IC50 = 15 nM T05409 CA04YQ 44267357 IC50 = 16 nM T05409 C3XA6O 44267359 IC50 = 11 nM T05409 CRKW25 44267368 IC50 = 3.5 nM T05409 CSDH98 44267369 IC50 = 2.4 nM T05409 CXQ13J 44273070 Ki = 23 nM T05409 CN7DR4 44275416 IC50 > 100000 nM T05409 C6I3TP 44275459 IC50 = 2300 nM T05409 C0D1BU 44275460 IC50 = 800 nM T05409 CBW4U8 44275461 IC50 = 300 nM T05409 CE48ZG 44275545 IC50 = 3000 nM T05409 CR78JL 44275546 IC50 = 1000 nM T05409 C1XW8V 44275712 IC50 = 4000 nM T05409 CMH8D4 44275713 IC50 > 100000 nM T05409 C6OJV1 44275764 IC50 > 60000 nM T05409 CH06AM 44275765 IC50 = 800 nM T05409 C7WDL8 44275775 IC50 = 10000 nM T05409 CYN0C4 44275794 IC50 = 10000 nM T05409 C54UHQ 44275795 IC50 > 60000 nM T05409 C7GH6B 44275869 IC50 = 15000 nM T05409 CDAN01 44275870 IC50 = 10000 nM T05409 CPNY12 44275871 IC50 > 100000 nM T05409 CSFD75 44275911 IC50 = 1200 nM T05409 CER04J 44275916 IC50 = 900 nM T05409 C1S6PA 44275933 IC50 = 800 nM T05409 CNFQ10 44275934 IC50 = 10000 nM T05409 C32HTK 44275937 IC50 = 3000 nM T05409 C4MR2S 44275948 IC50 = 300 nM T05409 CR4FL6 44283329 IC50 = 3.3 nM T05409 CFY54T 44283330 IC50 = 0.69 nM T05409 CBGP93 44283343 IC50 = 92 nM T05409 CN2X9D 44283344 IC50 = 218 nM T05409 CR81ZW 44283379 IC50 = 5.9 nM T05409 CCG20E 44283411 IC50 = 9.8 nM T05409 C5DR0V 44283412 IC50 = 7.4 nM T05409 C51YKA 44283534 IC50 = 3.2 nM T05409 CE7T1H 44283535 IC50 = 19 nM T05409 CAT9O4 44283552 IC50 = 122 nM T05409 CXD62O 44283599 IC50 = 763 nM T05409 CFD83W 44283893 IC50 = 58 nM T05409 C1XJ0W 44285058 IC50 = 4060 nM T05409 CHG51O 44285096 IC50 = 10000 nM T05409 CYT67M 44285121 IC50 = 9700 nM T05409 CFL9Y2 44285271 IC50 = 170 nM T05409 CN8Z4H 44295334 Ki = 0.7 nM T05409 C1K9TL 44295879 IC50 = 2.2 nM T05409 C7ZK6W 44295891 IC50 = 1.7 nM T05409 CSE6U2 44295892 IC50 = 2.4 nM T05409 CQ07SX 44295893 IC50 = 5.2 nM T05409 C3G2VM 44295920 IC50 = 865 nM T05409 C6Y1TE 44295939 IC50 = 7 nM T05409 C62VIB 44295941 IC50 = 1850 nM T05409 CDF39L 44295958 IC50 = 36 nM T05409 CFIG72 44295966 IC50 = 137 nM T05409 C6MXZ5 44295979 IC50 = 4260 nM T05409 C9F2HK 44296019 IC50 = 83 nM T05409 CD9M3U 44296036 IC50 = 118 nM T05409 C5Z6AR 44296037 IC50 = 1.2 nM T05409 CR1M7T 44303110 Ki = 24 nM T05409 CN5YE7 44305121 IC50 = 484 nM T05409 C35AID 44305131 IC50 = 1490 nM T05409 CEM4D9 44305132 IC50 = 1922 nM T05409 CVS47D 44305140 IC50 = 486 nM T05409 C5D2WT 44305173 IC50 = 140 nM T05409 C45NAZ 44305193 IC50 = 16 nM T05409 CCEN18 44305370 IC50 = 3 nM T05409 C97JBA 44305372 IC50 = 22 nM T05409 CYN2E6 44305391 IC50 = 55 nM T05409 CMC5H9 44314997 Ki = 330000 nM T05409 CLT0D3 44317068 Ki = 14000 nM T05409 CFQ3V4 44317087 Ki = 17000 nM T05409 CB9PO2 44324428 IC50 > 1000 nM T05409 CBF46I 44324644 IC50 = 226 nM T05409 C0Y8EC 44324645 IC50 = 73 nM T05409 CF9M7Y 44324653 IC50 > 1000 nM T05409 CK4R2O 44324830 IC50 = 735 nM T05409 C0O3FJ 44324831 IC50 = 165 nM T05409 C0A8MV 44324877 IC50 = 2 nM T05409 CP6K4X 44325010 IC50 = 12 nM T05409 C92CXR 44325039 IC50 = 1000 nM T05409 CJ6VC5 44325055 IC50 = 26 nM T05409 C9KD1P 44325081 IC50 = 48 nM T05409 C2ZG6V 44325082 IC50 = 20 nM T05409 CE0BW7 44325086 IC50 = 9 nM T05409 C6A1TX 44325087 IC50 = 35 nM T05409 CNHV10 44325092 IC50 = 35 nM T05409 C78HBX 44325093 IC50 = 37 nM T05409 CFNJ58 44325094 IC50 = 356 nM T05409 CDMZ17 44325095 IC50 > 1000 nM T05409 C1V3HD 44325102 IC50 = 200 nM T05409 CNT5D4 44325166 IC50 = 282 nM T05409 C0LH2X 44325169 IC50 = 338 nM T05409 C9ZX5S 44325207 IC50 = 171 nM T05409 CO0S6K 44325221 IC50 > 1000 nM T05409 C24XTA 44325222 IC50 = 47 nM T05409 CX70LB 44325223 IC50 = 34 nM T05409 CK4XN1 44325232 IC50 > 1000 nM T05409 C3J1QZ 44325246 IC50 > 1000 nM T05409 CAI35V 44325247 IC50 = 96 nM T05409 CMZY36 44325303 IC50 = 4 nM T05409 C10GFT 44329218 IC50 > 1000 nM T05409 C3VT0G 44329350 IC50 = 505 nM T05409 C3W8UX 44329454 IC50 > 1000 nM T05409 CMR38A 44329534 IC50 > 1000 nM T05409 CW2GK4 44344567 Ki = 2 nM T05409 C2EFO5 44364784 IC50 > 10000 nM T05409 CIG7T5 44364906 IC50 = 99 nM T05409 CF53QE 44364917 IC50 = 136 nM T05409 CG75AN 44377126 Ki = 1.1 nM T05409 CA3U8H 44386919 IC50 > 1000 nM T05409 CF2I3D 44388021 IC50 = 81900 nM T05409 C1FRV0 44400757 IC50 = 39200 nM T05409 CK79BM 44400838 IC50 > 100000 nM T05409 C8J4XB 44401169 IC50 > 100000 nM T05409 CFON28 44404945 IC50 = 0.08 nM T05409 C2PV3I 44404953 IC50 = 8 nM T05409 CAE21M 44413731 IC50 = 114 nM T05409 C9U1ZG 44413802 IC50 = 286 nM T05409 C90RTX 44413815 IC50 = 205 nM T05409 C04XPF 44422282 IC50 = 13.8 nM T05409 CLJN68 44422283 IC50 = 12.6 nM T05409 C06HJB 44446952 Ki = 27 nM T05409 CNK7X5 44446953 Ki = 5100 nM T05409 CEB78N 44446954 Ki = 950 nM T05409 CMO78A 44446956 Ki = 35 nM T05409 CV6H2M 44446957 Ki = 75 nM T05409 CF4KE1 44446959 Ki = 12 nM T05409 CW9C0E 44446960 Ki = 46 nM T05409 CQB5M0 44446963 Ki = 190 nM T05409 C94POY 44446965 Ki = 19 nM T05409 CBX2U9 44446967 Ki = 180 nM T05409 CRZ6B3 44446968 Ki = 79 nM T05409 CY9O4I 44446969 Ki = 10 nM T05409 C4PQ7D 44446970 Ki = 120 nM T05409 C96KIY 44446972 Ki = 37 nM T05409 CK1EM5 44446974 Ki = 300 nM T05409 C4V6RZ 44446975 Ki = 180 nM T05409 CBL9E6 44446976 Ki = 75 nM T05409 CVYX54 44446979 Ki = 640 nM T05409 CAI9Z6 44446980 Ki = 1500 nM T05409 C86KVP 44446984 Ki = 11000 nM T05409 C0GBP1 44454501 IC50 = 90 nM T05409 CND23X 44454625 IC50 = 36 nM T05409 CKO40E 44454648 IC50 = 5 nM T05409 C4XKJ6 44454674 IC50 = 19 nM T05409 C9O5YF 44454700 IC50 = 6 nM T05409 C18UOF 44454730 IC50 = 9 nM T05409 CAS59Y 44454780 IC50 = 8 nM T05409 CR32ML 44454831 IC50 = 6 nM T05409 C10OTH 44454833 IC50 = 2 nM T05409 CYK78A 44454905 IC50 = 19000 nM T05409 CSJ30Q 44454908 IC50 = 1540 nM T05409 CC2IS3 44454957 Ki = 1300 nM T05409 C1ESI2 44454959 Ki = 5.4 nM T05409 C8L0MV 44454960 Ki = 38 nM T05409 CBG6T0 44454987 Ki = 2.4 nM T05409 CN7UW3 44455013 Ki = 1.2 nM T05409 CC5L7S 44455015 Ki = 730 nM T05409 C6KDT1 44455016 Ki = 0.8 nM T05409 CF4ML7 44455018 Ki = 23 nM T05409 CZI6S1 44455047 Ki = 13 nM T05409 C3UF6E 44455406 Ki = 2.6 nM T05409 CJG71N 44455407 Ki = 140 nM T05409 C0IR5W 44455428 Ki = 130 nM T05409 C62KSV 44455429 Ki = 410 nM T05409 CR9WL2 44455430 Ki = 0.28 nM T05409 CRS9Q5 44458298 IC50 = 50 nM T05409 CS42ZF 44458316 IC50 = 4.5 nM T05409 C9WR8P 44460526 Ki > 100 nM T05409 C3OMR2 44460818 Ki = 408 nM T05409 CF31QH 44475015 IC50 = 63.1 nM T05409 CA1YC9 44626604 Ki = 130 nM T05409 CK6S5H 44626708 Ki = 1850 nM T05409 C0EJ1F 44626709 Ki = 68 nM T05409 CZR23J 44626710 Ki > 10000 nM T05409 CQB06H 44626711 Ki = 172 nM T05409 C17IGS 44627959 Ki = 2500 nM T05409 CM1DL3 44627960 Ki = 85 nM T05409 CNZ8L0 44628063 Ki > 5000 nM T05409 CRU86P 44628064 Ki > 10000 nM T05409 CS5BG9 44628065 Ki = 52 nM T05409 C65RAJ 45102601 IC50 = 0.631 nM T05409 CTOA14 45485236 Ki = 260 nM T05409 CS7F5N 49822299 IC50 = 6.9 nM T05409 CU1L9K 49822380 IC50 = 413 nM T05409 CYS2H7 49822381 IC50 = 4862 nM T05409 C1F3PN 53308743 IC50 = 1900 nM T05409 CN12AO 53353383 IC50 > 100000 nM T05409 C51GUC 53354365 IC50 > 100000 nM T05409 CRJ5P9 53354369 IC50 > 100000 nM T05409 C4G2HT 53354470 IC50 > 100000 nM T05409 CV19KH 54517870 IC50 = 0.8 nM T05409 CH5GT1 54580745 IC50 = 7 nM T05409 CV7D4R 54583711 IC50 = 22 nM T05409 C0PT5U 54583724 IC50 = 5 nM T05409 CSZW50 54583725 IC50 = 1.9 nM T05409 CI1Q0O 54584674 IC50 = 28 nM T05409 CF0EN3 54585609 IC50 = 20 nM T05409 CL1V8A 54585610 IC50 = 0.6 nM T05409 CJLW49 54585631 IC50 = 0.3 nM T05409 C4HPD3 54586623 IC50 = 4.8 nM T05409 CB9K6C 54586624 IC50 = 6 nM T05409 C8I6KJ 54587647 IC50 = 0.3 nM T05409 CGH0S7 54589400 IC50 > 100000 nM T05409 CDP80H 54751930 IC50 = 0.36 nM T05409 CFHP85 56646670 IC50 = 420 nM T05409 CZD09H 56668219 IC50 = 50000 nM T05409 CR3CQ0 56673957 IC50 = 9.7 nM T05409 CGF09H 56680595 IC50 = 430 nM T05409 C0J2DT 56683924 IC50 = 0.51 nM T05409 CF75JN 56953635 IC50 > 100000 nM T05409 CQ64IE 56953636 IC50 > 100000 nM T05409 C9RJF3 56953637 IC50 > 100000 nM T05409 CM7VP3 56953638 IC50 > 100000 nM T05409 C1BWY5 56953762 IC50 = 70000 nM T05409 C4VJI0 56953763 IC50 > 100000 nM T05409 C7JYZ1 56953764 IC50 > 100000 nM T05409 CH67KO 56953765 IC50 > 100000 nM T05409 CSW96U 56955172 IC50 = 48000 nM T05409 CFG17Q 56955173 IC50 = 30000 nM T05409 C76MEC 56955271 IC50 > 100000 nM T05409 CWGA37 56955272 IC50 > 100000 nM T05409 C28VDY 56955273 IC50 > 100000 nM T05409 C1QSV9 56955274 IC50 = 70000 nM T05409 CDU0R7 57335180 IC50 = 0.3 nM T05409 CA2Q7G 59607553 IC50 = 1500 nM T05409 CF62AH 59607562 IC50 = 5.4 nM T05409 CE9CM4 59607602 IC50 = 8 nM T05409 C4W2SP 59607629 IC50 = 4.5 nM T05409 CNZS03 59607667 IC50 = 25 nM T05409 C7S8YK 59607671 IC50 = 24 nM T05409 CP1KF2 59607681 IC50 = 26 nM T05409 CXV47G 59607684 IC50 = 21.3 nM T05409 C5CU7Y 59607693 IC50 = 44 nM T05409 C7LIU2 59607708 IC50 = 0.38 nM T05409 CR29JK 59607723 IC50 = 54 nM T05409 CL6S1A 59607741 IC50 = 1.5 nM T05409 CY4C8R 59607748 IC50 = 6.7 nM T05409 C74KMT 59607750 IC50 = 275 nM T05409 CX6B9A 59607793 IC50 = 60 nM T05409 CD56KW 59607797 IC50 = 1950 nM T05409 CG04FH 59607804 IC50 = 4182 nM T05409 CL2A6S 59607817 IC50 = 1370 nM T05409 C67VWG 59607853 IC50 = 111 nM T05409 C0D1QP 59607855 IC50 = 1.6 nM T05409 C49HEL 59607873 IC50 = 212 nM T05409 CCQ4T6 59607925 IC50 = 792 nM T05409 C7UTZ3 60182323 IC50 > 1000 nM T05409 C80FME 67362517 IC50 > 1000 nM T05409 CY1O5K 68749792 IC50 = 2 nM T05409 C64XBZ 70681347 IC50 > 70000 nM T05409 C4N3VW 70681348 IC50 > 100000 nM T05409 C5EHM1 70681503 IC50 > 100000 nM T05409 CFP12D 70683616 IC50 > 100000 nM T05409 CYVJ36 70683617 IC50 = 51000 nM T05409 CYD34L 70685541 IC50 = 12000 nM T05409 C1DZ3J 70685542 IC50 = 39000 nM T05409 C4BN0J 70689859 IC50 > 100000 nM T05409 CHM4W5 70692015 IC50 = 70000 nM T05409 CUX89K 70694685 Ki = 5.3 nM T05409 CFT06N 70696054 IC50 = 33000 nM T05409 C6MW3C 70696243 IC50 = 180000 nM T05409 C2IAG5 70696244 IC50 = 130000 nM T05409 C9P3EA 70696729 Ki = 1.6 nM T05409 CZSK89 71449083 IC50 = 12 nM T05409 CJ6T7O 71455231 IC50 = 27000 nM T05409 C0TGA7 71455232 IC50 < 60 nM T05409 CIPT41 71456155 IC50 > 1000 nM T05409 C4JK9N 71460699 IC50 = 300 nM T05409 CU73LD 71465043 IC50 = 3162.28 nM T05409 CH2Y7D 73671778 Ki = 36 nM T05409 CRXZ43 74223551 Ki = 20 nM T05409 C4VAC5 74223552 Ki = 52 nM T05409 CGQ57F 74223553 Ki = 32 nM T05409 CNW6S9 74223554 Ki = 36 nM T05409 C2O5QX 74223555 Ki = 9 nM T05409 CD3K9M 74223556 Ki = 29 nM T05409 C5RI6Y 74223618 Ki = 26 nM T05409 CU89YM 74223619 Ki = 470 nM T05409 C9VF7S 74223620 Ki = 86 nM T05409 CT9AW2 75031588 IC50 = 63.1 nM T05409 CK4O2F 87218352 IC50 = 1000 nM T05409 C8O1QX 87218371 IC50 = 630.96 nM T05409 C92GXJ 87218373 IC50 = 79.43 nM T05409 C8I9AL 87218397 IC50 = 1258.93 nM T05409 CUT8K1 87218444 IC50 = 39.81 nM T05409 C4BQD9 87218492 IC50 = 125.89 nM T05409 C8NEO1 87218514 IC50 = 31.62 nM T05409 CR45XW 87218658 IC50 = 125.89 nM T05409 C3OGP8 87218678 IC50 = 3.162 nM T05409 C0DUB7 87218698 IC50 = 3.162 nM T05409 C89OAU 87218826 IC50 = 630.96 nM T05409 C1UMO7 87218835 IC50 = 316.23 nM T05409 CLIT52 87218933 IC50 = 316.23 nM T05409 C2L9SX 87218987 IC50 = 1 nM T05409 CE09GY 87219028 IC50 = 1 nM T05409 CREO05 87219032 IC50 = 15.85 nM T05409 C4FML3 87219128 IC50 = 630.96 nM T05409 CM96JH 87219174 IC50 = 50.12 nM T05409 C1ON9G 90645547 Ki = 2.9 nM T05409 C6S0WK 90645548 Ki = 2.5 nM T05409 CS3FI2 90645549 Ki = 1.5 nM T05409 C59XED 90645550 Ki = 2 nM T05409 C8TK7S 90645551 Ki = 24 nM T05409 CNW3Y4 90645552 Ki = 8.2 nM T05409 C98ZFL 90645553 Ki = 44.1 nM T05409 CU8S4K 90645554 Ki = 59 nM T05409 CUD73A 90645555 Ki = 3.4 nM T05409 CK3S7U 90645556 Ki = 17.9 nM T05409 CQ87DK 90668200 IC50 = 79432.82 nM T05409 C1ZF3A 90668201 IC50 > 1000000 nM T05409 CCQ4Z7 90668202 IC50 > 1000000 nM T05409 CL2X3Z 90668203 IC50 > 1000000 nM T05409 C0WNR3 90668204 IC50 = 2511.89 nM T05409 C4HRO8 90668205 IC50 = 50118.72 nM T05409 CJG51C 90668206 IC50 > 1000000 nM T05409 CVH9P8 90668207 IC50 > 1000000 nM T05409 C83VPI 90668208 IC50 > 1000000 nM T05409 C54ESG 90668209 IC50 = 794.33 nM T05409 CX4MK8 90668210 IC50 > 1000000 nM T05409 CX5MA6 90668211 IC50 = 63.1 nM T05409 C3YZO5 90668278 IC50 = 6309.57 nM T05409 CWL1M3 122195270 IC50 > 100000 nM T05409 CN6UZ5 122195271 IC50 > 100000 nM T05409 C6CV7K 122195272 IC50 = 50000 nM T05409 CHE75Z 122195273 IC50 = 35000 nM T05409 C6RY2A 122195274 IC50 = 90000 nM T05409 C14TSF 122195275 IC50 > 100000 nM T05409 CIE12T 122195276 IC50 > 100000 nM T05409 C4DXT1 122195277 IC50 > 100000 nM T05409 CNV2J7 122195278 IC50 > 100000 nM T05409 CEQ47H 137631571 Ki = 49 nM T05409 CD4W3X 137635075 Ki = 1750 nM T05409 CES28O 137635451 Ki = 162 nM T05409 C8SO1T 137637613 Ki = 78 nM T05409 CF1K3S 137641249 Ki = 30 nM T05409 CHZ12D 137641745 Ki = 50 nM T05409 C0LGQ7 137642603 Ki = 4.2 nM T05409 C1NQ5R 137642653 Ki = 18 nM T05409 CIW5U3 137643490 Ki = 7 nM T05409 CR8MV2 137644362 Ki = 46 nM T05409 CO34MF 137645779 Ki = 252 nM T05409 C3CNQ2 137645957 Ki = 4.6 nM T05409 CS1E2Z 137650230 Ki > 0.00001 nM T05409 C4V2MU 137650778 Ki = 54 nM T05409 CI2H4K 137650843 Ki = 40 nM T05409 C52RST 137651616 Ki = 95 nM T05409 CRP35D 137651684 Ki = 12 nM T05409 CV39SO 137652265 Ki = 2 nM T05409 CYVE92 137652476 Ki = 22 nM T05409 CNR8J1 137654552 Ki = 61 nM T05409 CJLH69 137654770 Ki = 95 nM T05409 C8R7SP 137655314 Ki = 1650 nM T05409 CCTF28 137656413 Ki = 54 nM T05409 CC4BS6 137659320 Ki = 140 nM T05409 C0CAZ6 137661239 Ki = 260 nM T05409 C3W7NF 137661387 Ki = 61 nM T05409 CG6KB7 155512629 IC50 = 125.89 nM T05409 C9KP4F 155513439 IC50 = 1258.93 nM T05409 CPZI26 155513951 IC50 = 20 nM T05409 C1HOG5 155514738 IC50 = 1258.93 nM T05409 C7DQ3S 155516431 IC50 = 0.8 nM T05409 CN7Z5E 155516694 IC50 = 0.631 nM T05409 C21TUL 155520317 IC50 = 2.512 nM T05409 CX1YU9 155522135 IC50 = 1995.26 nM T05409 C30EFX 155523092 IC50 = 2511.89 nM T05409 C7WI9L 155526996 IC50 = 19.95 nM T05409 C1G7LY 155529942 IC50 = 39.81 nM T05409 CVXJ96 155533580 IC50 = 1 nM T05409 CNV2A8 155535176 IC50 = 398.11 nM T05409 CFM26N 155547799 IC50 = 79.43 nM T05409 C1RUT3 155552503 IC50 = 1 nM T05409 CUE8Y9 155557693 IC50 = 1995.26 nM T05409 CS7ZV8 155565351 IC50 = 7943.28 nM T05409 C0VK3G 44344579 Ki = 2 nM T05409 C2PVI1 44344594 Ki = 1.2 nM T05409 D02NQB 10430040 IC50 = 6 nM T05409 D04QJY 123982 Ki = 1.7 nM T05409 D07APP 131255 IC50 > 100000 nM T05409 D09NAJ 445114 IC50 = 30 nM T05409 D0B3UN 44580458 Ki > 100000 nM T05409 D0F8AR 45485268 Ki = 1.4 nM T05409 D0K1MA 9913857 IC50 = 6.9 nM T05409 D0N4RO 44377139 Ki = 1.3 nM T05409 D0N8YA 159596 IC50 = 50000 nM T05409 D0P4KL 135411330 IC50 > 100000 nM T05409 D0PB5Q 3132 IC50 = 1 nM T83797 CI7DT1 11857432 IC50 = 313 nM T83797 CHR92S 11858109 IC50 = 64 nM T83797 CDKH57 11858286 IC50 = 161 nM T83797 C4Z9CN 24769780 IC50 = 59 nM T70176 D04AIT 5280445 IC50 = 20000 nM T70176 D04LVK 57379345 IC50 = 3970 nM T70176 D05SBO 46220502 IC50 > 500 nM T70176 D07POC 176870 IC50 > 100000 nM T70176 D08CDI 208908 IC50 = 11000 nM T70176 D0AZ3C 5291 IC50 > 100000 nM T70176 D0E6XR 3062316 IC50 > 5000 nM T70176 D0EG1I 9926791 IC50 > 10000 nM T70176 D0K8KX 5280343 IC50 = 40000 nM T70176 D00RYA 16750271 IC50 = 7000 nM T70176 D00UZR 5330286 IC50 > 5000 nM T70176 D02NNV 3038525 IC50 > 5000 nM T70176 D02RJY 11442891 IC50 = 462 nM T70176 D02ZQS 16095342 IC50 = 3500 nM T70176 D03LWG 53235510 IC50 > 10000 nM T70176 D05ADP 160355 IC50 = 100 nM T70176 D06WHY 16747683 IC50 < 6 nM T70176 D07DTV 11338033 IC50 = 47 nM T70176 D07HPJ 11476171 IC50 > 10000 nM T70176 D08MXP 44631912 IC50 > 50000 nM T70176 D08UUL 46700756 IC50 > 10000 nM T70176 D0CY1B 6420138 Ki = 390 nM T70176 D0E3TC 44259 IC50 = 0.1 nM T70176 D0LF1U 5287969 Ki = 40 nM T70176 D0M0XB 10302451 IC50 = 10000 nM T70176 D0P0KN 16739650 IC50 = 3 nM T70176 D0Q7RE 16007391 Ki > 10000 nM T70176 D0Q9UX 16718576 IC50 = 45 nM T70176 D0S5RC 3025986 Ki = 38 nM T70176 D0Z1DH 10029385 IC50 = 2800 nM T70176 D0WS1V 448991 IC50 = 9 nM T70176 D0A3MV 448014 IC50 = 100000 nM T70176 D00BPA 4592 IC50 = 1200 nM T70176 D02YAQ 6603857 IC50 > 8000 nM T70176 D04FHB 6918852 Ki = 3 nM T70176 D0D3PX 46926350 IC50 = 1 nM T70176 D0F9WF 5459308 IC50 > 50000 nM T70176 D0L5YF 5329032 IC50 > 10000 nM T70176 D0Q7HO 4705 IC50 = 250000 nM T70176 D0U2TQ 644215 IC50 < 5.2 nM T70176 CS13FC 1941 IC50 = 25000 nM T70176 CRD89J 2236 IC50 > 20000 nM T70176 CJ17AM 4877 IC50 = 18000 nM T70176 C2BR0H 9221 IC50 = 185000 nM T70176 C08IAE 10143 IC50 > 50000 nM T70176 CA6YG7 10153 IC50 > 50000 nM T70176 C97TNH 10177 IC50 = 2200 nM T70176 CG3YN1 10215 IC50 = 70000 nM T70176 CGO94B 34458 IC50 > 50000 nM T70176 CW67XG 65275 IC50 > 100000 nM T70176 C63WLY 89644 IC50 > 10 ug.mL-1 T70176 CDJN90 96710 IC50 = 1200 nM T70176 CC50TS 101300 IC50 > 50000 nM T70176 C5JE2Z 104860 IC50 > 10 ug.mL-1 T70176 C0T7KS 108168 IC50 > 20000 nM T70176 CT1M8Y 119204 IC50 > 50000 nM T70176 CS74HZ 145726 IC50 > 500000 nM T70176 CT5SN2 145826 IC50 = 4000 nM T70176 C3F0HX 148297 IC50 = 15000 nM T70176 C1WV7B 148745 IC50 = 15000 nM T70176 C28CSW 158883 IC50 = 35 nM T70176 CI1NA5 159926 IC50 > 10 ug.mL-1 T70176 CZCL56 159999 IC50 > 50000 nM T70176 CO28NX 160500 IC50 > 50000 nM T70176 CF34UR 160501 IC50 > 50000 nM T70176 C6X3QK 161218 IC50 = 25000 nM T70176 CW9UP3 165274 IC50 = 30000 nM T70176 CL9I8P 167493 IC50 > 20000 nM T70176 CYBA43 177458 IC50 > 10 ug.mL-1 T70176 CLC05O 272989 IC50 > 10000 nM T70176 CLW30H 314123 IC50 = 1300 nM T70176 CIXA81 316313 IC50 = 1026000 nM T70176 CHO64G 378604 IC50 > 500000 nM T70176 CA19KV 378607 IC50 = 760000 nM T70176 COYB64 379086 IC50 = 1230000 nM T70176 C4J8QT 383495 IC50 = 11000 nM T70176 C0ZJ4O 398147 IC50 > 10000 nM T70176 CU1TA8 398149 IC50 > 100000 nM T70176 C29RZS 405795 IC50 = 330 nM T70176 CX31DW 405797 IC50 = 570 nM T70176 CKU63M 405799 IC50 = 820 nM T70176 C5B2AG 405898 IC50 = 16000 nM T70176 C6YIR0 405899 IC50 > 28000 nM T70176 CT0UZ6 405900 IC50 > 28000 nM T70176 C3MS5E 405913 IC50 = 24000 nM T70176 C2R7KY 405914 IC50 = 24000 nM T70176 CTW50F 405915 IC50 = 11000 nM T70176 C0O3AP 405916 IC50 > 28000 nM T70176 C1Q3TV 405917 IC50 = 15000 nM T70176 CR15WE 405963 IC50 > 28000 nM T70176 CI7D3Y 406259 IC50 = 15000 nM T70176 COL36P 406261 IC50 = 23000 nM T70176 C4MNG8 445840 IC50 = 440 nM T70176 CPRG75 447446 IC50 = 540 nM T70176 CNF1P5 447652 IC50 = 2900 nM T70176 C69SAW 447766 IC50 = 12 nM T70176 CJA3D4 447958 Ki = 290 nM T70176 CFDR89 447959 Ki = 60 nM T70176 CXS8U2 447960 Ki = 70 nM T70176 CB9F1O 447961 Ki = 2 nM T70176 C6A3LY 447962 Ki = 220 nM T70176 C1ZG2U 449087 IC50 = 37 nM T70176 CFHO09 481744 IC50 > 200000 nM T70176 CNVT43 481745 IC50 > 200000 nM T70176 CM7NF4 481746 IC50 > 200000 nM T70176 CL15VX 481748 IC50 > 200000 nM T70176 CVN83J 656950 IC50 > 10000 nM T70176 CW12BK 657138 IC50 = 1500 nM T70176 CE73JV 819275 IC50 = 370 nM T70176 C6C2PK 832258 IC50 = 55110 nM T70176 C8YC3Z 1187348 IC50 = 105100 nM T70176 C9THB6 2495235 IC50 < 10000 nM T70176 CHC5I0 2971839 IC50 > 10000 nM T70176 CE4TS0 3000629 IC50 = 6800 nM T70176 CPOJ12 3078519 IC50 = 30 nM T70176 C2Z8DX 3084007 IC50 > 20000 nM T70176 CCN9D5 3142817 IC50 = 700 nM T70176 C4ELP8 3160258 IC50 = 690 nM T70176 C4CA5U 3323623 IC50 = 46 nM T70176 C9Z7AU 3496894 IC50 = 300 nM T70176 CHGS79 3551941 IC50 = 60 nM T70176 C1D2PA 3803479 IC50 > 10000 nM T70176 C4ZT3K 4155347 IC50 = 80 nM T70176 C2GZP6 4247366 IC50 = 1499.68 nM T70176 C7WXK1 4469813 IC50 = 35000 nM T70176 CAXZ94 4475481 IC50 = 1000 nM T70176 C4DU1B 4475482 IC50 = 38000 nM T70176 CN95RS 4477128 IC50 = 560 nM T70176 CAD5G8 4477129 IC50 = 5.7 nM T70176 C7NTG0 4477130 IC50 = 8.9 nM T70176 C0WHD7 4477131 IC50 = 1000 nM T70176 CK3XT1 4477132 IC50 = 660 nM T70176 CFEU51 4478473 IC50 = 3000 nM T70176 CU1N7T 5287990 IC50 = 59 nM T70176 C4R7SZ 5288222 IC50 = 3 nM T70176 C15WJX 5288527 IC50 = 1 nM T70176 C4MUT0 5289179 IC50 = 324 nM T70176 CHK2V0 5289411 IC50 = 34 nM T70176 C8A1SH 5319404 IC50 > 15000 nM T70176 CX74MR 5319620 IC50 = 2150 nM T70176 CEJ0C2 5327664 IC50 = 1410 nM T70176 C3L4MH 5329496 IC50 = 49000 nM T70176 CMVG29 5329578 IC50 = 13000 nM T70176 CZG0R9 5329598 IC50 = 59000 nM T70176 CCK8Q5 5329599 IC50 = 2900 nM T70176 CFB24A 5329600 IC50 = 500 nM T70176 CMTY12 5329601 IC50 = 220 nM T70176 CS3CM2 5329602 IC50 = 120 nM T70176 CFQ5N9 5329603 IC50 = 1.1 nM T70176 CTC68O 5329656 IC50 = 46 nM T70176 C2Q7FO 5329713 IC50 = 3930 nM T70176 CM9V8E 5329715 IC50 = 2110 nM T70176 C8BXI6 5329717 IC50 = 6590 nM T70176 C9X0YE 5329718 IC50 = 1070 nM T70176 C54EYJ 5329719 IC50 = 40400 nM T70176 CW0Z9J 5329753 IC50 = 13 nM T70176 C4GPF6 5329921 IC50 = 20 nM T70176 CBW30C 5330047 IC50 = 8 nM T70176 CGI90W 5330278 IC50 = 439 nM T70176 CL5I2U 5330279 IC50 = 230 nM T70176 C4V5QX 5330356 IC50 > 360 nM T70176 C5TGL0 5330583 IC50 = 78 nM T70176 CK4CO2 5330614 IC50 = 122 nM T70176 CJI2G7 5330615 IC50 = 102 nM T70176 CH4IV5 5330616 IC50 = 91 nM T70176 C8LTE0 5330617 IC50 = 68 nM T70176 CFD3I6 5330618 IC50 = 121 nM T70176 CE2X0C 5330619 IC50 = 214 nM T70176 CE4I0K 5330620 IC50 = 26 nM T70176 C96AEG 5330621 IC50 = 29 nM T70176 CLXG43 5330622 IC50 = 95 nM T70176 C16LYJ 5330623 IC50 = 46 nM T70176 C3VZF8 5330624 IC50 = 33 nM T70176 C48LEV 5330625 IC50 = 63 nM T70176 CD6Y7M 5330626 IC50 = 896 nM T70176 C5LVY9 5330627 IC50 = 1691 nM T70176 CFXB43 5330628 IC50 = 1927 nM T70176 C2CV3M 5330629 IC50 = 428 nM T70176 CF6TG7 5330630 IC50 = 1068 nM T70176 CGSQ67 5330631 IC50 = 1294 nM T70176 C5HTQ4 5330632 IC50 = 603 nM T70176 CWM6X8 5330633 IC50 = 2171 nM T70176 CP5CX4 5330634 IC50 = 53 nM T70176 C73DEJ 5330636 IC50 = 547 nM T70176 C7K9LJ 5330637 IC50 = 1711 nM T70176 CJK60U 5330638 IC50 = 2538 nM T70176 CQ14LV 5330639 IC50 = 52 nM T70176 CKFY92 5330641 IC50 = 812 nM T70176 C6ROJ7 5330642 IC50 = 160 nM T70176 CK9SR7 5330717 IC50 = 1610 nM T70176 C28WYZ 5330718 IC50 < 60 nM T70176 C3U0TG 5330830 IC50 = 500 nM T70176 CL1FH5 5330832 IC50 = 180 nM T70176 C1P2ZA 5330847 IC50 = 84 nM T70176 CPTX95 5330921 IC50 = 1200 nM T70176 CM7YU9 5330940 IC50 = 1999.86 nM T70176 CY8I9S 5330941 IC50 > 10000 nM T70176 CTP59F 5330943 IC50 = 960 nM T70176 CJY53K 5330945 IC50 = 2600.16 nM T70176 CLX0N2 5330946 IC50 = 83.95 nM T70176 CM98LE 5330947 IC50 = 6000 nM T70176 C7F3VU 5330948 IC50 = 2500 nM T70176 CU2J0N 5330949 IC50 = 36.98 nM T70176 CDGU09 5330954 IC50 = 170 nM T70176 CO47PT 5330955 IC50 = 2 nM T70176 C74POB 5330957 IC50 = 454.99 nM T70176 CZLM34 5330958 IC50 = 2 nM T70176 C92JWU 5330964 IC50 = 8500 nM T70176 C34KCE 5330965 IC50 = 16.98 nM T70176 CN82AU 5330966 IC50 = 2500 nM T70176 CP7R3A 5330967 IC50 = 20 nM T70176 CTG4R2 5330970 IC50 = 79.98 nM T70176 C82XZJ 5330971 IC50 > 10000 nM T70176 CS2J6E 5330972 IC50 = 223.87 nM T70176 CA2C9J 5330973 IC50 = 34 nM T70176 CDAO37 5330974 IC50 = 84.92 nM T70176 C2DP5F 5330975 IC50 = 705 nM T70176 C3ZM9T 5330976 IC50 = 164.82 nM T70176 CBOR85 5330977 IC50 = 68 nM T70176 CJUN-60 5330978 IC50 = 990 nM T70176 C2L8UJ 5330979 IC50 = 1000 nM T70176 C2PUK5 5330980 IC50 = 599.79 nM T70176 CP0XM5 5330981 IC50 = 500 nM T70176 CWP3K6 5330982 IC50 = 1499.68 nM T70176 C8MZ9P 5330983 IC50 = 1000 nM T70176 CIK65Y 5330984 IC50 > 10000 nM T70176 CGUS16 5330985 IC50 > 10000 nM T70176 C9ZRT7 5330986 IC50 = 82.99 nM T70176 CLE4S2 5330987 IC50 = 89.95 nM T70176 CL7NW9 5330988 IC50 = 50 nM T70176 C8K3XT 5330989 IC50 = 10000 nM T70176 CS13AI 5330990 IC50 = 5997.91 nM T70176 C09MCN 5330991 IC50 = 629.51 nM T70176 CUS65V 5330992 IC50 = 650 nM T70176 CT12DK 5330993 IC50 = 199.99 nM T70176 CXVQ32 5330995 IC50 > 10000 nM T70176 CAW94B 5330996 IC50 > 10000 nM T70176 CZ1U9Q 5330997 IC50 > 10000 nM T70176 C7LE5C 5330998 IC50 = 47.97 nM T70176 CYDL73 5330999 IC50 = 74 nM T70176 CD5K9H 5331000 IC50 = 29 nM T70176 CY0L5X 5331002 IC50 = 67 nM T70176 CFNO38 5331003 IC50 = 56 nM T70176 CS3A8F 5331081 IC50 = 40 nM T70176 CG4W8K 5331082 IC50 = 4 nM T70176 CD4C2A 5331083 IC50 = 12 nM T70176 C6AT8V 5331084 IC50 = 64 nM T70176 CJVS23 5331085 IC50 = 33 nM T70176 CZ29FN 5331086 IC50 = 4 nM T70176 CYL78A 5331087 IC50 = 82 nM T70176 CJ87XR 5331088 IC50 = 88 nM T70176 CFB3K7 5331089 IC50 = 190 nM T70176 C9WY1O 5331090 IC50 = 270 nM T70176 C9ZK3D 5331091 IC50 = 30 nM T70176 C6RJC8 5331092 IC50 = 9 nM T70176 C0IOY8 5331093 IC50 = 1500 nM T70176 CMD08O 5331094 IC50 > 10000 nM T70176 CMDK89 5331095 IC50 = 250 nM T70176 C6LC4P 5331096 IC50 = 9 nM T70176 C8BK2Z 5331097 IC50 = 68 nM T70176 C0IC6Z 5331098 IC50 = 68 nM T70176 CHO5J2 5331099 IC50 = 300 nM T70176 CD6YO5 5331100 IC50 = 530 nM T70176 C6FU8S 5331101 IC50 = 340 nM T70176 C1Y0NB 5331102 IC50 = 49 nM T70176 CQV6P8 5331103 IC50 = 5700 nM T70176 CLJ1W5 5332196 IC50 = 1.1 ug.mL-1 T70176 CDQ3M7 5359485 IC50 = 3.3 ug.mL-1 T70176 C54BYP 5360741 IC50 = 3.6 ug.mL-1 T70176 CY7P2R 5408233 IC50 > 50000 nM T70176 CKT4I5 5473014 IC50 = 400 nM T70176 C5JZ1X 5473015 IC50 = 23000 nM T70176 C36XBW 5714753 IC50 > 20 ug.mL-1 T70176 C9E5NV 5828196 IC50 = 27000 nM T70176 C3BH0S 6538740 IC50 = 680 nM T70176 CCRM28 6538898 IC50 = 1280 nM T70176 C0O8DH 6538899 IC50 = 3970 nM T70176 CW9S3K 6538900 IC50 = 310 nM T70176 C5Y7MX 6538901 IC50 = 30 nM T70176 CZH30S 6538902 IC50 = 2980 nM T70176 CK4HA1 6538931 IC50 > 100000 nM T70176 C3SVJ4 6538972 IC50 = 93000 nM T70176 C0N8IC 6538973 IC50 = 39000 nM T70176 C0R3HT 6538974 IC50 = 24000 nM T70176 C1JPE7 6538975 IC50 > 100000 nM T70176 C91GSM 6538976 IC50 = 95000 nM T70176 CD4ZY6 6538977 IC50 = 28000 nM T70176 C4KO2H 6538978 IC50 = 85000 nM T70176 C59NXD 6538979 IC50 = 25000 nM T70176 C18DCI 6538980 IC50 = 22000 nM T70176 CJMA92 6538981 IC50 = 1000 nM T70176 CQU63M 6538982 IC50 = 5000 nM T70176 CR62XM 6538983 IC50 = 19000 nM T70176 C2HZQ7 6538984 IC50 > 100000 nM T70176 C9XQV0 6538985 IC50 = 32000 nM T70176 CEG54P 6538986 IC50 = 7000 nM T70176 C4APW5 6538987 IC50 = 6000 nM T70176 C48ERS 6538988 IC50 = 7000 nM T70176 CFA5Z0 6538989 IC50 = 4000 nM T70176 CA68PN 6538990 IC50 = 15000 nM T70176 C8YH9W 6538991 IC50 = 5000 nM T70176 C6V0LQ 6538992 IC50 = 18000 nM T70176 C76LEK 6538993 IC50 = 36000 nM T70176 CBO5S8 6538994 IC50 = 26000 nM T70176 C4D0WX 6538995 IC50 = 2000 nM T70176 CS6DQ2 6538996 IC50 = 5000 nM T70176 CH04KA 6538997 IC50 = 1000 nM T70176 CRH42M 6538998 IC50 = 700 nM T70176 CZ2PE0 6538999 IC50 = 2000 nM T70176 CXW9Y6 6539000 IC50 = 3000 nM T70176 C8CSQ3 6539001 IC50 > 10000 nM T70176 CU8PL7 6539002 IC50 = 12000 nM T70176 CH70WZ 6539003 IC50 = 8000 nM T70176 CXF78K 6539004 IC50 > 10000 nM T70176 C3E2VM 6539005 IC50 = 500 nM T70176 CK7O9B 6539006 IC50 = 200 nM T70176 C6R2TO 6539007 IC50 = 95000 nM T70176 CZ7F0B 6539008 IC50 > 10000 nM T70176 CWP7M9 6539009 IC50 = 36 nM T70176 CT9XA5 6539010 IC50 = 10 nM T70176 C1MGU7 6539011 IC50 < 3 nM T70176 C6MDN7 6539012 IC50 > 100000 nM T70176 C47VIS 6539013 IC50 > 100000 nM T70176 CS8VA4 6539014 IC50 > 100000 nM T70176 C2Z8SX 6539015 IC50 = 81000 nM T70176 C04YNQ 6539016 IC50 = 22000 nM T70176 C5WK8I 6539017 IC50 = 6 nM T70176 CS6VL5 6539018 IC50 = 4000 nM T70176 CM94KT 6539019 IC50 = 8800 nM T70176 CN9T5R 6539020 IC50 = 150 nM T70176 CDC73B 6539021 IC50 = 620 nM T70176 C26JOQ 6539022 IC50 < 3 nM T70176 CY3Q5G 6539023 IC50 = 5 nM T70176 CCA1U5 6539024 IC50 < 3 nM T70176 C09UJZ 6539025 IC50 < 12 nM T70176 C0L5BW 6539026 IC50 = 4 nM T70176 CW9MN4 6539027 IC50 = 5 nM T70176 C3NZ8V 6539028 IC50 < 3 nM T70176 C5UKP1 6539029 IC50 = 5 nM T70176 C4Q3PB 6539030 IC50 < 3 nM T70176 CK2O8A 6539031 IC50 < 3 nM T70176 CT3WD6 6539032 IC50 > 10000 nM T70176 COW18E 6539033 IC50 < 3 nM T70176 C97DGO 6539034 IC50 < 3 nM T70176 CHZ3C2 6539035 IC50 < 3 nM T70176 CM18AC 6539036 IC50 = 16 nM T70176 CKT59A 6539038 IC50 < 3 nM T70176 COXM80 6539040 IC50 = 8 nM T70176 C6MRY3 6539278 Ki > 20000 nM T70176 CXQ92S 6539279 Ki > 20000 nM T70176 CEL82X 6539280 Ki = 80 nM T70176 CU2N3Q 6539281 Ki > 20000 nM T70176 CN1AU7 6539282 Ki = 670 nM T70176 C6IB7U 6539283 Ki = 2500 nM T70176 CC62GN 6539284 Ki = 1200 nM T70176 C0J8QA 6539285 Ki = 100 nM T70176 CR8KA0 6539286 Ki = 40 nM T70176 C9P5OX 6539287 Ki > 20000 nM T70176 C3KM1T 6539288 Ki > 20000 nM T70176 C8OC9M 6539289 Ki = 110 nM T70176 C7IWS5 6539290 Ki > 10000 nM T70176 CM35CV 6539291 Ki = 140 nM T70176 CT7MP9 6539292 Ki = 30 nM T70176 C1CRW6 6539293 Ki = 110 nM T70176 C3HQ1G 6539294 Ki > 20000 nM T70176 CQ9U3J 6539295 Ki = 60 nM T70176 COL0X2 6539296 Ki = 800 nM T70176 CKV60H 6539297 Ki = 160 nM T70176 CBC56F 6539298 Ki > 20000 nM T70176 C0LMW1 6539299 Ki = 4100 nM T70176 C51VJH 6539300 Ki = 400 nM T70176 C0K1VF 6539301 Ki = 300 nM T70176 C95ETX 6539302 Ki = 20 nM T70176 CY03LO 6539303 Ki = 100 nM T70176 CO8NR2 6539304 Ki = 700 nM T70176 CN76AU 6539305 Ki = 50 nM T70176 C6UZF0 6539306 Ki = 140 nM T70176 C84MNG 6539307 Ki = 50 nM T70176 C38NYA 6539308 Ki = 50 nM T70176 C08SLD 6539309 Ki = 30 nM T70176 C6VB9U 6539310 Ki = 130 nM T70176 CB6N1Y 6539311 Ki = 90 nM T70176 CKJW72 6539312 Ki = 100 nM T70176 CQV1J5 6539313 Ki = 80 nM T70176 C1M4LA 6539314 Ki = 30 nM T70176 CO4QV9 6539315 Ki = 360 nM T70176 C96XMO 6539316 Ki = 270 nM T70176 CM2N8O 6539359 Ki = 5 nM T70176 CTD0X9 6539360 Ki = 19900 nM T70176 CUK02R 6539362 Ki = 1 nM T70176 CZY97M 6539363 IC50 = 3 nM T70176 C9X8DW 6539364 Ki = 10 nM T70176 CM9FT4 6539365 Ki = 150 nM T70176 C9Y3KC 6539366 Ki = 150 nM T70176 C6Z0WU 6539368 Ki = 10 nM T70176 CY1W7D 6539369 Ki = 6 nM T70176 CO3A4B 6539370 IC50 = 1.995 nM T70176 C8RND3 6539371 Ki = 6 nM T70176 CB69DA 6539372 Ki = 1 nM T70176 CL18KE 6539373 Ki = 10 nM T70176 C74TAS 6539375 Ki = 10 nM T70176 C2GFT6 6539376 Ki = 10 nM T70176 C7SHN5 6539377 Ki = 1 nM T70176 CQM14U 6539378 Ki = 310 nM T70176 CTBE09 6539379 Ki = 3 nM T70176 CWN7Q3 6539380 Ki = 8 nM T70176 CN2XV5 6539381 Ki = 160 nM T70176 C5TC2D 6539382 Ki = 1990 nM T70176 C8KT3B 6539383 Ki = 1260 nM T70176 CQ84MY 6539384 Ki = 60 nM T70176 C5Z4AQ 6539385 Ki = 190 nM T70176 CZQ56A 6539386 Ki = 500 nM T70176 CA5YC3 6539387 Ki = 20 nM T70176 C6A0FQ 6539388 Ki = 190 nM T70176 CX0T4J 6539389 Ki = 790 nM T70176 C7E2ZP 6539390 Ki > 19950 nM T70176 CAP2D7 6539391 Ki > 19950 nM T70176 CYC62P 6539392 Ki = 100 nM T70176 C9NC7H 6539393 Ki = 50 nM T70176 C4R2HQ 6539394 Ki = 190 nM T70176 CU85HS 6539395 Ki = 20 nM T70176 CQ51SX 6539396 Ki = 6 nM T70176 CFVB56 6539397 Ki = 2500 nM T70176 C8K7LC 6539398 Ki > 19950 nM T70176 C6K7UA 6539399 Ki = 3980 nM T70176 C5U4AD 6539400 Ki > 19950 nM T70176 CO04SD 6539401 Ki > 19950 nM T70176 CC0Q9Z 6539402 Ki > 19950 nM T70176 C5S6FX 6539403 Ki > 19950 nM T70176 CNR94M 6539404 Ki > 19950 nM T70176 CVD04S 6539405 Ki > 19950 nM T70176 C3BCG6 6539406 Ki > 19950 nM T70176 CEV0Q5 6539407 Ki > 19950 nM T70176 C9PRY5 6539408 Ki > 19950 nM T70176 C1L3BI 6539409 Ki > 19950 nM T70176 C72GAY 6539410 Ki > 19950 nM T70176 CZ67GY 6539411 Ki > 19950 nM T70176 C9G2CO 6539412 Ki > 19950 nM T70176 C9VEJ5 6539413 Ki > 19950 nM T70176 CF9AB1 6539414 Ki > 19950 nM T70176 C5TUV1 6539415 Ki > 19950 nM T70176 CCES70 6539416 Ki > 19950 nM T70176 CWAN68 6539417 Ki > 19950 nM T70176 CXI64Y 6539418 Ki > 19950 nM T70176 C97DXU 6539419 Ki > 19950 nM T70176 CO39EQ 6539420 Ki > 19950 nM T70176 C7A1QZ 6539421 Ki > 19950 nM T70176 CA04MW 6539422 Ki > 19950 nM T70176 CG5ZY9 6539423 Ki > 19950 nM T70176 C92LYE 6539424 Ki > 19950 nM T70176 CU9A6K 6539425 Ki > 19950 nM T70176 C2FUA0 6539426 Ki > 19950 nM T70176 CD4Z7F 6539427 Ki > 19950 nM T70176 CG6C5K 6539428 Ki > 19950 nM T70176 CPS9K1 6539429 Ki > 19950 nM T70176 C9JW4Z 6539430 Ki > 19950 nM T70176 C6NW0F 6539431 Ki > 19950 nM T70176 CK0MH3 6539432 Ki > 19950 nM T70176 C35HXQ 6539433 Ki > 19950 nM T70176 C0RS9Q 6539434 Ki > 19950 nM T70176 CWZE47 6539435 Ki > 19950 nM T70176 CIRF95 6539436 Ki > 19950 nM T70176 C6RIL5 6539437 Ki = 5000 nM T70176 CCEB18 6539438 Ki > 19950 nM T70176 C9FRV1 6539439 Ki > 19950 nM T70176 CS1K9T 6539440 Ki > 19950 nM T70176 CD26TN 6539441 Ki > 19950 nM T70176 C6U4BK 6539442 Ki > 19950 nM T70176 CPU3R1 6539443 Ki > 19950 nM T70176 CP36QM 6539444 Ki > 19950 nM T70176 CQ39BD 6539445 Ki = 3980 nM T70176 CJO9W0 6539446 Ki > 19950 nM T70176 C7X8AJ 6539447 Ki > 19950 nM T70176 C1LV4T 6539448 Ki > 19950 nM T70176 C7M9VJ 6539449 Ki > 19950 nM T70176 CP7J3S 6539569 IC50 = 62 nM T70176 C7C9BO 6539578 IC50 > 1000 nM T70176 CCXU69 6539586 IC50 = 341 nM T70176 CQTU34 6539587 IC50 = 484 nM T70176 COI57D 6539588 IC50 = 639 nM T70176 CQ97IV 6539591 IC50 > 1000 nM T70176 C70OTV 6539592 IC50 > 1000 nM T70176 CAI54V 6539593 IC50 > 1000 nM T70176 C9ABL1 6539595 IC50 > 1000 nM T70176 C87GNI 6539596 IC50 > 1000 nM T70176 CGO8A0 6539597 IC50 > 1000 nM T70176 C4TJI2 6539598 IC50 > 1000 nM T70176 CHWL84 6539599 IC50 > 1000 nM T70176 C6P4BO 6539600 IC50 > 1000 nM T70176 CG1C4I 6539601 IC50 > 1000 nM T70176 CHP97J 6539602 IC50 > 1000 nM T70176 C79LMV 6539603 IC50 > 1000 nM T70176 CDS2B8 6539604 IC50 > 1000 nM T70176 CWJ6C1 6539605 IC50 > 1000 nM T70176 CNV39L 6539606 IC50 > 1000 nM T70176 CH54ZS 6539607 IC50 > 1000 nM T70176 C14VJA 6539608 IC50 = 497 nM T70176 C1M3ZI 6539609 IC50 = 631 nM T70176 C7U2TC 6539610 IC50 > 1000 nM T70176 C5XBK1 6539611 IC50 > 1000 nM T70176 CNE0Y5 6539612 IC50 > 1000 nM T70176 CK3W6M 6539613 IC50 > 1000 nM T70176 CJV73P 6539614 IC50 > 1000 nM T70176 C1PVJ8 6539615 IC50 > 1000 nM T70176 C60GSI 6539616 IC50 = 10 nM T70176 C3LX4A 6539618 IC50 = 0.34 nM T70176 CK4D8T 6539619 IC50 = 24.5 nM T70176 CN91SM 6539620 IC50 = 9.1 nM T70176 C7DR8V 6539621 IC50 = 10.7 nM T70176 CA5EJ9 6539622 IC50 = 61.6 nM T70176 C0FZA1 6539623 IC50 = 10.7 nM T70176 CVK3F7 6539624 IC50 = 23.4 nM T70176 C95NAZ 6539625 IC50 = 602 nM T70176 CT5S9Y 6539626 IC50 = 871 nM T70176 CS9BC8 6539627 IC50 = 17.4 nM T70176 C2MBR7 6539628 IC50 > 2000 nM T70176 C1T0IC 6539629 IC50 = 407 nM T70176 C43SPU 6539630 IC50 = 0.33 nM T70176 CFC9K7 6539631 IC50 = 490 nM T70176 CLE6A4 6539632 IC50 = 166 nM T70176 CNFV70 6539738 IC50 > 19000 nM T70176 CBRC53 6539739 IC50 > 20000 nM T70176 C8QG1T 6539740 IC50 > 21000 nM T70176 CW7VD6 6539741 IC50 > 20000 nM T70176 C5UFS1 6539742 IC50 > 19000 nM T70176 C5XSJ6 6539743 IC50 > 19000 nM T70176 CRL2P4 6539744 IC50 > 20000 nM T70176 CSWR78 6539745 IC50 > 20000 nM T70176 CXI8M7 6539746 IC50 > 21000 nM T70176 CSZF21 6539747 IC50 > 21000 nM T70176 CFM2K9 6539748 IC50 > 20000 nM T70176 C1QFC6 6539749 IC50 > 21000 nM T70176 CFQ5R7 6539750 IC50 > 20000 nM T70176 C0R6WV 6539751 IC50 > 21000 nM T70176 C25FMB 6539752 IC50 > 19000 nM T70176 CRB1O3 6539753 IC50 = 440 nM T70176 CZ17AH 6539754 IC50 > 19000 nM T70176 CT4K0Z 6539755 IC50 > 20000 nM T70176 CMIS20 6539756 IC50 > 20000 nM T70176 CTNR52 6539757 IC50 > 19000 nM T70176 CJ58QK 6539758 IC50 = 450 nM T70176 CJ4U3H 6610355 IC50 = 8000 nM T70176 CVU8N0 6918710 IC50 = 120 nM T70176 CFYE71 9341021 IC50 = 3000 nM T70176 CJ1ML3 9412007 IC50 = 3000 nM T70176 C31XGW 9825189 IC50 = 7 nM T70176 CNZD42 9836341 IC50 = 12 nM T70176 C81KXQ 9837883 IC50 = 204 nM T70176 CZ9MB2 9843864 Ki = 597 nM T70176 CXQ9J0 9856983 Ki > 5000 nM T70176 C41QWA 9857146 IC50 > 10000 nM T70176 C1UCQ8 9858505 IC50 = 18 nM T70176 CV3Q7H 9858586 IC50 = 3 nM T70176 CRC65X 9863786 IC50 > 25000 nM T70176 CW8V0K 9864418 IC50 > 20000 nM T70176 CM5Z8X 9869943 IC50 > 1000 nM T70176 CSL50Q 9886746 IC50 = 230 nM T70176 CXA5C8 9893493 IC50 > 50000 nM T70176 C2Y3WG 9907612 IC50 = 55 nM T70176 C7JGW4 9910100 IC50 = 190 nM T70176 CQ8P1R 9921498 IC50 = 376 nM T70176 CYBJ50 9921823 IC50 = 18 nM T70176 C08OBL 9922207 IC50 = 77 nM T70176 CYW49X 9927718 IC50 > 25000 nM T70176 CTV25B 9934643 IC50 = 20900 nM T70176 CQD2W7 9935079 IC50 = 992 nM T70176 CS5KX9 9938299 IC50 > 10000 nM T70176 CIR5D1 9944548 IC50 = 54 nM T70176 C6L0SN 9946036 IC50 = 28 nM T70176 CJO47T 9948405 IC50 > 10000 nM T70176 C57URF 9951265 IC50 = 36 nM T70176 CD5M3J 9952008 IC50 = 140 nM T70176 C41HSX 9965506 IC50 = 72 nM T70176 CLG32N 9967203 IC50 = 14 nM T70176 CV28XH 9979332 IC50 = 2100 nM T70176 CTU1O9 9979700 Ki = 7 nM T70176 C37GXK 9983303 IC50 > 20000 nM T70176 CHFO23 9994136 IC50 > 200000 nM T70176 CDHT89 9999155 Ki = 327 nM T70176 CV8I5X 9999342 IC50 > 10000 nM T70176 CPSY37 10001536 IC50 = 3 nM T70176 CCQ5A6 10023782 Ki = 1756 nM T70176 CVE1W8 10024433 Ki = 432 nM T70176 CYT3Z6 10045499 Ki = 2166 nM T70176 C7YD1X 10048045 IC50 > 25000 nM T70176 CT70MI 10049465 IC50 = 6000 nM T70176 CICK35 10066656 IC50 = 5 nM T70176 C18DAI 10069391 Ki = 886 nM T70176 C1JUF8 10073832 IC50 > 50000 nM T70176 C2C1BP 10089048 IC50 > 20000 nM T70176 C93UVK 10092544 IC50 = 3600 nM T70176 CZP6U0 10110571 IC50 = 7 nM T70176 C50QLR 10110675 IC50 = 9 nM T70176 C7TA9J 10113568 IC50 = 17782.79 nM T70176 CXBW34 10114553 IC50 = 14 nM T70176 C0H9JX 10125875 IC50 = 1000 nM T70176 CTXW95 10126509 IC50 = 100 nM T70176 CH8UX5 10132679 IC50 = 127 nM T70176 CGT4F0 10134861 IC50 = 20 nM T70176 CL2F5J 10135889 IC50 = 10 nM T70176 CPT91S 10138993 IC50 = 30 nM T70176 CZJI60 10141037 IC50 > 10000 nM T70176 C94WRY 10143231 IC50 > 10000 nM T70176 C08VYL 10158127 IC50 = 10 nM T70176 C69DHW 10158652 IC50 < 16000 nM T70176 C79SUC 10158868 IC50 = 4 nM T70176 C68GUB 10159114 IC50 = 20 nM T70176 C59FGN 10165455 IC50 = 490 nM T70176 CQG5R4 10173796 IC50 = 4 nM T70176 CC78NE 10179293 IC50 = 711 nM T70176 CLE8V6 10182312 IC50 = 7 nM T70176 C5Y9PK 10183407 IC50 = 75 nM T70176 CW2Y7N 10200092 IC50 = 16 nM T70176 CIGT47 10202305 IC50 = 9 nM T70176 CVRO56 10204194 IC50 = 7 nM T70176 C5P8JC 10206423 IC50 = 2439 nM T70176 COWF65 10215271 IC50 = 0.3 nM T70176 C4JW0S 10221609 IC50 = 48 nM T70176 CHM97B 10221628 IC50 = 10 nM T70176 C84VWO 10221806 IC50 = 250 nM T70176 CLW0H7 10223662 IC50 = 10 nM T70176 CTS43G 10238877 IC50 > 25000 nM T70176 CH48JA 10239038 IC50 = 450 nM T70176 C5TQ7X 10247543 IC50 > 10000 nM T70176 C1KX3P 10248401 Ki = 1039 nM T70176 CE19JD 10249602 Ki = 3137 nM T70176 CB2GC4 10250350 IC50 = 4 nM T70176 CJ1AN4 10251513 Ki = 51 nM T70176 C0NMU1 10267663 IC50 = 62 nM T70176 CTMH81 10268741 IC50 = 65 nM T70176 C0Z8JG 10269818 IC50 = 23 nM T70176 C7XRU0 10270270 IC50 = 294 nM T70176 CS3MR8 10270322 IC50 = 18 nM T70176 CG65JV 10275574 IC50 = 22 nM T70176 CJGH26 10275985 IC50 = 19500 nM T70176 C8GJ9A 10286242 IC50 = 1000 nM T70176 CWB04N 10291997 IC50 = 15 nM T70176 C58NEO 10295144 IC50 = 1400 nM T70176 C85MHR 10297090 IC50 = 40 nM T70176 C6PL7N 10297469 IC50 = 30 nM T70176 C6J7FS 10297929 IC50 = 1700 nM T70176 C8RD3V 10301884 IC50 > 10000 nM T70176 CKA8B0 10308522 IC50 = 2 nM T70176 COD9W2 10308706 IC50 = 40 nM T70176 C6S9AO 10310395 IC50 = 230 nM T70176 CKNL70 10319097 Ki = 24 nM T70176 C9J3RM 10320107 Ki = 297 nM T70176 C6USY4 10339994 IC50 = 30 nM T70176 CMY9D2 10340715 Ki = 151 nM T70176 C2BW1Y 10352920 IC50 = 7000 nM T70176 CVN8T9 10379252 IC50 = 1300 nM T70176 CC3L8Z 10430000 Ki = 156 nM T70176 C62KGB 10430385 IC50 = 11000 nM T70176 CTJ8K5 10430386 IC50 = 24000 nM T70176 CFNM76 10434333 Ki = 495 nM T70176 CHB2D8 10449125 Ki = 6266 nM T70176 CB86LA 10456600 IC50 = 3.4 nM T70176 C2WQ8M 10473563 IC50 > 10000 nM T70176 C7PLI5 10478569 IC50 > 50000 nM T70176 CRX6F0 10479082 IC50 > 20000 nM T70176 CXCO41 10479319 Ki = 2 nM T70176 CQ24PL 10503846 IC50 = 20000 nM T70176 C21BTO 10524103 IC50 > 100000 nM T70176 CWYE93 10615524 IC50 = 900 nM T70176 CW2K9B 10634429 IC50 = 2400 nM T70176 C7MJ0P 10807095 IC50 = 200 nM T70176 C4VX1Q 11065484 IC50 = 690 nM T70176 CJ7U4I 11161778 IC50 = 16000 nM T70176 C94QUD 11163861 Ki = 10 nM T70176 CEW9U5 11173394 IC50 = 500000 nM T70176 CQ6J7A 11210632 IC50 = 350 nM T70176 C35SDM 11219672 IC50 > 500000 nM T70176 C2W5RC 11235063 IC50 > 100000 nM T70176 C30PKR 11248978 IC50 = 5300 nM T70176 C69HPR 11257553 Ki = 149 nM T70176 CW76SZ 11265905 IC50 = 200000 nM T70176 C18OKN 11266386 IC50 > 500000 nM T70176 CB32AD 11268094 IC50 = 140 nM T70176 C3N1MF 11270500 IC50 = 17 nM T70176 C6C3JX 11281930 IC50 > 10000 nM T70176 CHB2U6 11284129 IC50 = 16 nM T70176 CBOP58 11293798 Ki > 10000 nM T70176 CSXY78 11294864 IC50 = 5400 nM T70176 C3UKE2 11300307 IC50 = 400000 nM T70176 CNT19Q 11315446 IC50 = 8 nM T70176 C2X7TJ 11316094 IC50 < 3 nM T70176 CPU9I3 11316975 IC50 = 2100 nM T70176 CMXI90 11324412 Ki > 2500 nM T70176 CQ8I4H 11328863 IC50 = 3400 nM T70176 C26BZX 11362471 Ki = 5760 nM T70176 CG1T5J 11386640 IC50 = 10 nM T70176 CWXB93 11397177 Ki > 10000 nM T70176 C4EA5U 11403673 IC50 = 430000 nM T70176 C7AI2V 11432911 IC50 > 50000 nM T70176 CKU8Y3 11442383 IC50 = 6 nM T70176 C64IGY 11448608 Ki > 5000 nM T70176 CVN1C0 11477611 IC50 = 11 nM T70176 C6M9NC 11477626 IC50 > 50000 nM T70176 C9LA1E 11486283 IC50 = 574 nM T70176 CXT91K 11488074 IC50 = 260 nM T70176 C7G4VM 11508924 IC50 = 3 nM T70176 C3D9OU 11509538 IC50 = 57 nM T70176 CCX5Y9 11509539 IC50 = 17 nM T70176 CL1WN3 11518075 IC50 = 36 nM T70176 CU79NQ 11524833 IC50 = 17 nM T70176 C1RCA9 11525251 IC50 = 120 nM T70176 CL7X4Q 11530963 IC50 = 6900 nM T70176 C0X2AS 11533897 IC50 = 118 nM T70176 CR53ZL 11537871 IC50 = 8 nM T70176 CJIW92 11539281 IC50 = 35 nM T70176 CTG83F 11539329 Ki > 8600 nM T70176 CJ8BQ6 11552741 IC50 = 41 nM T70176 CCLR26 11552773 IC50 < 1 nM T70176 CVS32L 11560956 IC50 = 551 nM T70176 C1W5OC 11562531 IC50 = 247 nM T70176 C45QDX 11568147 IC50 = 50 nM T70176 C72XAP 11569937 IC50 = 62 nM T70176 CD3E8M 11574606 IC50 = 350 nM T70176 C9EIF4 11582467 IC50 = 24 nM T70176 CMIL86 11590363 Ki > 8600 nM T70176 C2V0DP 11598432 IC50 = 71 nM T70176 CPO6F9 11610059 IC50 = 521000 nM T70176 CSM62L 11626920 IC50 > 30000 nM T70176 CGX96V 11626927 IC50 > 30000 nM T70176 CTL6H8 11630942 IC50 > 35000 nM T70176 C95RDI 11631662 IC50 = 3 nM T70176 CIWA03 11632150 Ki = 239 nM T70176 CK34LS 11632737 IC50 > 10000 nM T70176 CABL68 11639899 IC50 = 72 nM T70176 C9T6SC 11640926 Ki > 8600 nM T70176 CEV5X2 11646645 Ki = 32 nM T70176 C2CVI7 11647020 Ki = 463 nM T70176 CCH38R 11654950 IC50 = 70 nM T70176 CQKD95 11669987 IC50 = 1 nM T70176 C9G3OH 11675718 IC50 = 19 nM T70176 COEL03 11676096 IC50 = 323 nM T70176 CYM9A8 11678367 IC50 = 266 nM T70176 CJ9KN7 11683817 IC50 > 10000 nM T70176 C1XYK2 11717025 IC50 = 3 nM T70176 C93KHF 11718021 Ki = 256 nM T70176 C9UA2S 11718220 IC50 > 250000 nM T70176 C28TNJ 11722322 IC50 > 200000 nM T70176 CR93CE 11743030 Ki = 13 nM T70176 CJSV21 11744184 Ki = 3967 nM T70176 CS36BH 11843159 IC50 > 40000 nM T70176 CW3K2L 11957417 IC50 = 1584.89 nM T70176 C6N0RY 11974955 Ki > 10000 nM T70176 CNIK34 11974956 Ki > 10000 nM T70176 C0YX7V 11974957 Ki > 10000 nM T70176 CLTK95 11975073 Ki = 84 nM T70176 CDP24B 11975074 Ki = 451 nM T70176 CXR6J8 11975075 Ki = 15 nM T70176 C2QV6O 11975201 Ki > 10000 nM T70176 CAP2M7 11975202 Ki > 10000 nM T70176 C5XWU4 11975203 Ki = 5141 nM T70176 CZF8T4 11975204 Ki > 10000 nM T70176 CX2AS7 11975205 Ki = 2030 nM T70176 C3OHQ1 11975206 Ki = 6 nM T70176 CSI4K0 12187419 IC50 = 1160000 nM T70176 C7PN1U 12187420 IC50 = 985000 nM T70176 CV6Z3P 12187421 IC50 = 951000 nM T70176 CB84XP 12187422 IC50 = 790000 nM T70176 C72HOU 12187423 IC50 = 1030000 nM T70176 CM6FE5 12187424 IC50 = 910000 nM T70176 CJR7W4 13521419 IC50 = 25000 nM T70176 C2Z8DQ 14624081 IC50 = 220 nM T70176 C86VOB 14887322 IC50 > 15000 nM T70176 C32LMH 15751152 IC50 = 940000 nM T70176 CP5AC1 15942652 IC50 = 87 nM T70176 CFPW41 16007116 Ki > 8600 nM T70176 C7BS2R 16037674 IC50 > 10000 nM T70176 CB2H4D 16037675 IC50 = 1700 nM T70176 C9TU1O 16046126 IC50 = 3.4 nM T70176 C3GY9M 16050532 Ki < 100 nM T70176 C8VL6K 16050623 Ki < 100 nM T70176 CCU4S2 16050624 Ki < 100 nM T70176 CPX83C 16050724 Ki < 100 nM T70176 C0Y4WS 16050816 Ki < 100 nM T70176 CSN3C9 16050817 Ki = 140 nM T70176 CZHJ34 16058637 IC50 = 2700 nM T70176 C7Z4LV 16095343 IC50 = 7000 nM T70176 C15QAG 16113377 IC50 = 2 nM T70176 C5GZ4J 16113378 IC50 = 2 nM T70176 C1O9SF 16113484 IC50 = 2 nM T70176 C0C5AZ 16129582 IC50 = 1517 nM T70176 CDO7W8 16202256 Ki = 1160 nM T70176 CU56EW 16664858 IC50 > 10000 nM T70176 C0H8UN 16730109 IC50 > 10000 nM T70176 CSE35D 16739464 IC50 = 320 nM T70176 C20OFQ 16739508 IC50 = 1600 nM T70176 C0TMW8 16739778 IC50 = 150 nM T70176 CCP56J 16739905 IC50 = 710 nM T70176 CQ64XI 16739921 IC50 = 330 nM T70176 CM3UF8 16739935 IC50 = 8600 nM T70176 CFEP56 16739948 IC50 = 22 nM T70176 C23KZR 16739951 IC50 = 420 nM T70176 C5UY9I 16741552 IC50 = 1840 nM T70176 CYQ9W5 16741728 IC50 = 32000 nM T70176 C9OQ1G 16750272 IC50 = 680 nM T70176 CW2SY5 16750291 IC50 = 2900 nM T70176 CIX7U2 16750304 IC50 > 10000 nM T70176 C6A3XS 16750306 IC50 = 6800 nM T70176 CB2TK1 16750327 IC50 > 10000 nM T70176 CH4O1C 16750328 IC50 = 3200 nM T70176 C90MJD 16750331 IC50 = 200 nM T70176 CCF2B3 17933136 IC50 = 68 nM T70176 C59CVU 19689599 IC50 = 8.9 nM T70176 C6H0EI 19754146 IC50 = 28500 nM T70176 CJC5F3 20741385 Ki = 2452 nM T70176 CH4B5K 21081523 IC50 > 5000 nM T70176 C25UKC 21081761 IC50 > 1000 nM T70176 CA61QF 21083895 IC50 = 31000 nM T70176 C78DCI 21680138 IC50 > 35000 nM T70176 C6WDM7 22099513 IC50 = 2100 nM T70176 C8YF5D 22099524 IC50 = 2110 nM T70176 C9RUO2 22273524 IC50 = 8 nM T70176 CUBY98 22273530 IC50 < 3 nM T70176 C31XZM 22273548 IC50 = 11 nM T70176 C71MEZ 22971096 IC50 = 50 nM T70176 CVX45U 22994151 IC50 = 2000 nM T70176 C9QLP0 23133323 IC50 > 20000 nM T70176 CG9HS7 23586143 IC50 = 1800 nM T70176 C42OBN 23586145 IC50 = 11000 nM T70176 CN39TP 23586146 IC50 = 730 nM T70176 CPL7J5 23635674 IC50 = 3 nM T70176 C63ROA 23645085 IC50 > 1000 nM T70176 CXYO32 23645086 IC50 = 5500 nM T70176 C6GP0X 23645088 IC50 = 124 nM T70176 C1BCP7 23645089 IC50 = 5 nM T70176 C0O2WB 23645090 IC50 = 7 nM T70176 CL2T3I 23645566 IC50 = 4 nM T70176 C16MYH 23645567 IC50 = 8 nM T70176 CV3Q1Z 23645568 IC50 = 61 nM T70176 CR53PW 23645569 IC50 = 92 nM T70176 CM20NA 23645570 IC50 = 17 nM T70176 CMJ4C7 23645571 IC50 = 2100 nM T70176 CBK47A 23645572 IC50 = 1200 nM T70176 CR5I7U 23645573 IC50 = 1200 nM T70176 CE7QN6 23645574 IC50 = 2 nM T70176 C8H2FO 23645576 IC50 = 7400 nM T70176 C6YF5D 23645577 IC50 = 400 nM T70176 C9G5EQ 23645578 IC50 = 270 nM T70176 C95CXB 23645579 IC50 = 120 nM T70176 CHK57M 23645580 IC50 = 250 nM T70176 CG3VB6 23646578 IC50 = 169 nM T70176 CG6D4M 23647319 IC50 > 10000 nM T70176 CY8Z7X 23647330 IC50 > 10000 nM T70176 C4XD8H 23647348 IC50 > 10000 nM T70176 CHI9J4 23654066 IC50 > 25000 nM T70176 C4KT2G 23654071 IC50 = 138 nM T70176 C3JWK1 23654166 IC50 = 185 nM T70176 CV8I2B 23654167 IC50 = 285 nM T70176 CU1M0Q 23654255 IC50 > 1000 nM T70176 C8N4DL 23654256 IC50 > 10000 nM T70176 CDON60 23654258 IC50 > 2000 nM T70176 CY7P0K 23654341 IC50 > 2000 nM T70176 C35HDM 23654345 IC50 = 276 nM T70176 C4TOU0 23654594 IC50 = 15.4 nM T70176 CG03YM 23654922 IC50 = 12.4 nM T70176 C2RV3U 24180608 IC50 > 30000 nM T70176 CA3I4T 24753787 IC50 > 50000 nM T70176 C7YG1N 24759534 IC50 = 12 nM T70176 CI70UD 24765900 Ki = 1800 nM T70176 C0VZQ5 24765998 IC50 = 450 nM T70176 C60JXM 24780352 IC50 = 2 nM T70176 CLBP72 24798571 IC50 > 10000 nM T70176 CCP2M3 24822704 IC50 > 50000 nM T70176 CI5B6S 24825779 IC50 > 50000 nM T70176 CZ48LS 24825971 IC50 > 50000 nM T70176 C61KPI 24856363 IC50 > 20000 nM T70176 CAZ15Y 24864077 IC50 = 850 nM T70176 CMG5W6 24864078 IC50 = 140 nM T70176 CFH3X8 24864079 IC50 = 3 nM T70176 CFK2B9 24882503 IC50 > 10000 nM T70176 C43HWQ 24883287 IC50 > 10000 nM T70176 C8DA5Q 24883334 IC50 > 10000 nM T70176 C13QYB 24884503 IC50 > 2000 nM T70176 CYDU89 24884773 IC50 = 13 nM T70176 CE2MR9 24884776 IC50 = 36 nM T70176 C8PD7V 24884981 IC50 = 15 nM T70176 CJH19T 24894883 IC50 = 42000 nM T70176 CB5TP8 24894992 IC50 = 23000 nM T70176 CFW40U 24894997 IC50 = 20000 nM T70176 CWV98O 24899557 IC50 = 77 nM T70176 CN13JF 24899915 IC50 = 0.84 ug.mL-1 T70176 CBWR97 24899916 IC50 = 2.4 ug.mL-1 T70176 C9F2JD 24899917 IC50 > 10 ug.mL-1 T70176 C64MTI 24900160 IC50 > 10 ug.mL-1 T70176 CO2I6Q 24900161 IC50 > 10 ug.mL-1 T70176 CLZ23U 24951610 IC50 > 30000 nM T70176 C7N4DI 24959043 IC50 > 100000 nM T70176 C6CVK4 24959046 IC50 > 100000 nM T70176 CB0V4I 24963033 IC50 = 1 nM T70176 CYK63A 24971312 IC50 = 1500 nM T70176 CMDB40 24971313 IC50 = 30 nM T70176 C60TVS 24971314 IC50 = 85000 nM T70176 C10QFL 24971315 IC50 = 730 nM T70176 CYCK73 24971316 IC50 = 1600 nM T70176 CPTJ24 24971317 IC50 = 90 nM T70176 CH58OF 24971318 IC50 = 25 nM T70176 CKDJ21 24971319 IC50 = 12 nM T70176 C5XZ0P 24971320 IC50 = 19 nM T70176 C43NMJ 24971321 IC50 = 38 nM T70176 CO5LI2 24971322 IC50 = 750 nM T70176 CF0QM6 24971323 IC50 = 110 nM T70176 C8CO4B 24971342 IC50 = 110 nM T70176 CAC94U 24991573 IC50 = 1070 nM T70176 CS3Q8B 24995659 Ki > 4000 nM T70176 CBK82P 25011729 IC50 = 17600 nM T70176 CP9WY7 25022741 IC50 = 736000 nM T70176 C7HD3I 25026174 Ki = 200 nM T70176 CSH7B8 25026574 Ki = 900 nM T70176 CB53EO 25026772 Ki = 900 nM T70176 C18LDH 25026775 Ki = 10000 nM T70176 C6N7KR 25032700 IC50 = 540 nM T70176 CX1HL8 25032704 Ki > 8570 nM T70176 C2ICS7 25065806 IC50 > 1000 nM T70176 C2KY1G 25094210 IC50 = 2273 nM T70176 CQ67BO 25113172 Ki > 3330 nM T70176 COV8Z0 25143021 IC50 > 10000 nM T70176 C6BWZ8 25145145 IC50 > 100 nM T70176 C78YWA 25145716 IC50 > 500 nM T70176 CI0E2L 25154395 IC50 = 270 nM T70176 CL1W5D 25154436 IC50 = 3900 nM T70176 CID5O7 25169255 Ki > 5000 nM T70176 CN2B0H 25169256 Ki > 5000 nM T70176 C4BV0K 25169528 IC50 = 5 nM T70176 CE65CO 25169529 IC50 = 20 nM T70176 CQ04LW 25171665 IC50 = 50 nM T70176 CU9KV5 25171666 IC50 = 30 nM T70176 CNJH95 25175218 IC50 = 348 nM T70176 C53JCN 25175220 IC50 = 4630 nM T70176 CP28KV 25176840 IC50 = 18 nM T70176 C4NBG3 25178327 IC50 = 4300 nM T70176 C85KCS 25178328 IC50 = 5300 nM T70176 C1VH9P 25178329 IC50 = 6800 nM T70176 CX0O5A 25178331 IC50 = 5100 nM T70176 CWZ61J 25178538 IC50 = 7700 nM T70176 CIG4H0 25178539 IC50 = 3600 nM T70176 C4GI6J 25178540 IC50 = 6300 nM T70176 CI39OW 25190761 IC50 = 40 nM T70176 C6M2HV 25190763 IC50 = 220 nM T70176 CX4Z1H 25195254 IC50 = 20 nM T70176 C6FGQ1 25206346 IC50 > 10000 nM T70176 CN5E0F 25263283 IC50 = 23000 nM T70176 CC71QJ 27666048 IC50 > 100000 nM T70176 CLX89Z 31940930 IC50 = 406000 nM T70176 CU53WB 42596953 IC50 = 920 nM T70176 CIDU19 42625518 IC50 = 44400 nM T70176 CM5QJ4 42628077 IC50 > 16000 nM T70176 CU9E4P 42629114 IC50 > 10000 nM T70176 CJ5U1X 42639664 IC50 > 10 ug.mL-1 T70176 CT27FZ 42642931 IC50 = 250 nM T70176 C30BQP 42642932 IC50 = 14000 nM T70176 C74LQM 42642933 IC50 = 180 nM T70176 CO42DC 44138048 IC50 > 10000 nM T70176 CL65QV 44138049 IC50 > 10000 nM T70176 C1IYU0 44139710 IC50 > 16000 nM T70176 C04IJO 44139711 IC50 = 3200 nM T70176 CLW80F 44160269 IC50 = 17000 nM T70176 C8KNA3 44219632 Ki > 4000 nM T70176 C0VIX4 44219633 Ki = 3100 nM T70176 CK73NR 44219749 IC50 > 50000 nM T70176 C6G2EC 44232693 IC50 = 1053 nM T70176 CFVC13 44232694 IC50 = 45 nM T70176 CV0FL9 44232695 IC50 = 14 nM T70176 CN0UM6 44232696 IC50 = 137 nM T70176 C4KUD5 44232697 IC50 = 29 nM T70176 CA05LE 44232698 IC50 = 55 nM T70176 CYCX40 44232939 IC50 = 160 nM T70176 CT1CU7 44232940 IC50 = 220 nM T70176 C4NW9L 44232941 IC50 = 83 nM T70176 CCG09Z 44235884 IC50 = 3900 nM T70176 CY8A7D 44235885 IC50 = 2 nM T70176 CE42KQ 44235886 IC50 = 1 nM T70176 C5R4QP 44235887 IC50 = 24 nM T70176 CLB67D 44235888 IC50 = 17 nM T70176 C2GRK8 44236107 IC50 = 31 nM T70176 C4AJ7M 44236108 IC50 = 248 nM T70176 CR27YG 44236109 IC50 = 47 nM T70176 CBN34C 44236110 IC50 = 59 nM T70176 CS8XM3 44236111 IC50 = 36 nM T70176 CZIT93 44236112 IC50 = 59 nM T70176 C09YHS 44236349 IC50 = 35 nM T70176 C13QXB 44236351 IC50 = 2 nM T70176 CJ37DI 44236353 IC50 = 19 nM T70176 CK5CF7 44236354 IC50 = 74 nM T70176 CMSW41 44361566 IC50 > 200000 nM T70176 C9M3GP 44361567 IC50 > 200000 nM T70176 CSBC59 44396134 IC50 > 20000 nM T70176 CO13WA 44397218 IC50 = 984 nM T70176 CZ18LR 44397301 IC50 = 462 nM T70176 C54JRW 44399701 IC50 = 43 nM T70176 CS9GM3 44400429 IC50 = 1000 nM T70176 C8L5ZH 44401437 IC50 = 2 nM T70176 CAN72B 44408691 IC50 = 26000 nM T70176 CWM75V 44412739 IC50 = 140 nM T70176 C5HZF2 44413509 IC50 = 14 nM T70176 C3D4FG 44413527 IC50 = 270 nM T70176 CFED20 44415457 IC50 = 140 nM T70176 C02ZHB 44432199 IC50 = 630 nM T70176 C4GYR5 44432201 IC50 = 1600 nM T70176 C87CHD 44432203 IC50 = 3000 nM T70176 CY0BU7 44432204 IC50 = 2600 nM T70176 C9LKR5 44432206 IC50 = 640 nM T70176 CM4Z3J 44432208 IC50 = 1600 nM T70176 CLG4J3 44432213 IC50 = 4400 nM T70176 CAX8F5 44440161 IC50 = 412 nM T70176 CK9H1G 44440214 IC50 = 10000 nM T70176 CDF70Q 44440215 IC50 = 605 nM T70176 CK8L4U 44440216 IC50 = 4443 nM T70176 CM2E3N 44440217 IC50 = 4219 nM T70176 CWL30H 44440218 IC50 = 10000 nM T70176 C6RD3G 44440219 IC50 = 2483 nM T70176 C52CDB 44440221 IC50 = 555 nM T70176 C2OC7L 44440222 IC50 > 10000 nM T70176 CFZS24 44440223 IC50 = 1264 nM T70176 CSA87R 44440224 IC50 = 612 nM T70176 CH76CV 44440225 IC50 = 123 nM T70176 CP80UK 44440226 IC50 = 4358 nM T70176 CFI06W 44440227 IC50 = 5281 nM T70176 CKSO82 44440228 IC50 = 2672 nM T70176 C8HWI1 44440229 IC50 = 1126 nM T70176 CVD97U 44440230 IC50 = 1895 nM T70176 C1B0TO 44440234 IC50 = 6652 nM T70176 CS5PY4 44440235 IC50 > 10000 nM T70176 C9AV4C 44440236 IC50 > 10000 nM T70176 C4Y8XV 44446930 IC50 = 180 nM T70176 CWBV18 44446940 IC50 = 520 nM T70176 CPR51F 44446941 IC50 = 230 nM T70176 CPW34M 44447902 IC50 = 500 nM T70176 C4V7JK 44447903 IC50 = 200 nM T70176 COZM30 44447904 IC50 = 1800 nM T70176 CX5ZB9 44447905 IC50 > 100000 nM T70176 CX5TI8 44447906 IC50 = 170 nM T70176 CQ7Y1B 44447907 IC50 = 7100 nM T70176 CB9RV2 44447912 IC50 = 10 nM T70176 C4MQJ7 44447913 IC50 = 24 nM T70176 C2N6CE 44447930 IC50 = 10 nM T70176 CLI16E 44465026 IC50 = 110 nM T70176 CQEM30 44480711 Ki = 16 nM T70176 CK1Q4M 44481490 Ki = 240 nM T70176 C8G3YW 44481491 Ki = 210 nM T70176 C53EDG 44481492 Ki > 4000 nM T70176 C4WHX7 44481494 Ki = 69 nM T70176 CRC7Y6 44481495 Ki = 41 nM T70176 C6MCD5 44481764 Ki = 450 nM T70176 CNFT56 44481765 Ki = 250 nM T70176 CRIB07 44481766 Ki = 138 nM T70176 C24AMY 44481768 Ki = 140 nM T70176 C1XA5C 44481769 Ki = 57 nM T70176 C8LN2S 44482036 Ki < 100 nM T70176 CD3YS7 44482037 Ki = 1100 nM T70176 C8MEU4 44482038 Ki = 290 nM T70176 CDOZ57 44482040 Ki = 150 nM T70176 CBJ8U7 44482041 Ki = 76 nM T70176 CX5W3P 44482303 Ki = 316 nM T70176 CKS3B9 44482304 Ki = 642 nM T70176 CNZ38Y 44482305 Ki = 209 nM T70176 C1O8SQ 44482306 Ki = 170 nM T70176 CJ56HF 44482307 Ki > 2500 nM T70176 C4WRN5 44541014 IC50 = 35.5 nM T70176 C3VRO9 44557921 IC50 > 10000 nM T70176 CWN43A 44562683 IC50 = 6 nM T70176 CE7LN0 44562736 IC50 = 4 nM T70176 C6PJI0 44562737 IC50 < 1 nM T70176 C8C6AW 44562738 IC50 = 2 nM T70176 C2HJ9Z 44563066 IC50 = 17 nM T70176 C83CZN 44563067 IC50 = 2 nM T70176 C28ZHE 44563068 IC50 = 56 nM T70176 C2J0WX 44563069 IC50 = 42 nM T70176 CSB8O2 44563070 IC50 = 2 nM T70176 CF0GM9 44563109 IC50 = 81 nM T70176 CUC3E6 44563110 IC50 = 62 nM T70176 C97AJO 44563111 IC50 < 1 nM T70176 CL3MW0 44563112 IC50 = 2 nM T70176 C1VQ2B 44563116 IC50 = 9 nM T70176 CP5GJ1 44563117 IC50 = 37 nM T70176 CSJ14N 44563119 IC50 = 15 nM T70176 CXEW65 44563120 IC50 = 3 nM T70176 C51TLU 44563144 IC50 < 1 nM T70176 CNR1B2 44563145 IC50 = 6 nM T70176 C0D1LO 44563146 IC50 < 1 nM T70176 CS19XE 44563151 IC50 = 11 nM T70176 C5VQG1 44563155 IC50 = 17 nM T70176 CK4GU3 44563156 IC50 = 95 nM T70176 CNS69D 44563157 IC50 = 14 nM T70176 CKU49O 44563158 IC50 = 140 nM T70176 CJV9S8 44563177 IC50 = 2 nM T70176 CV90NH 44563178 IC50 = 9 nM T70176 CK8F3Q 44563194 IC50 = 36 nM T70176 CH48EY 44563195 IC50 = 200 nM T70176 CXH34K 44563822 IC50 = 4 nM T70176 CLCH53 44563836 IC50 = 8.995 nM T70176 CQF3K1 44563837 IC50 = 3 nM T70176 CCP2E4 44570694 IC50 = 60 nM T70176 C9GU6J 44578536 IC50 < 3 nM T70176 CN41KS 44578537 IC50 = 24 nM T70176 CBNM35 44578538 IC50 = 8 nM T70176 CJZ04U 44578568 IC50 = 3 nM T70176 C05UQI 44578569 IC50 < 3 nM T70176 CD1U2S 44578570 IC50 < 3 nM T70176 C1MC0I 44578615 IC50 = 3 nM T70176 CFAW91 44578616 IC50 < 3 nM T70176 CYPJ70 44578617 IC50 = 17 nM T70176 CR0F7I 44578649 IC50 = 16 nM T70176 CZ57CL 44578651 IC50 = 9 nM T70176 C6ME2I 44578692 IC50 = 0.5 nM T70176 CQW72F 44578693 IC50 > 0.3 nM T70176 CA0HO5 44578694 IC50 = 46 nM T70176 C7Q1VU 44580077 IC50 > 20000 nM T70176 CL90SE 44580358 IC50 > 20000 nM T70176 CK1VE7 44580420 IC50 > 20000 nM T70176 CH2R7X 44580449 IC50 > 20000 nM T70176 C1VH0C 44580532 IC50 > 20000 nM T70176 CXC52J 44580649 IC50 > 20000 nM T70176 CE32BQ 44580689 IC50 > 20000 nM T70176 C8Z5AX 44580778 IC50 > 20000 nM T70176 C5I3HT 44580807 IC50 = 3 nM T70176 CMH2A3 44580824 IC50 = 16 nM T70176 CTP7I4 44580861 IC50 = 40 nM T70176 C4W9HX 44580967 IC50 = 229 nM T70176 CSE67T 44581007 IC50 = 168 nM T70176 CB0F8O 44581008 IC50 = 7 nM T70176 CKU1P7 44581009 IC50 = 158 nM T70176 C2ZIH5 44581010 IC50 = 28 nM T70176 C9HAU7 44581033 IC50 = 9 nM T70176 CL6Y9J 44581034 IC50 = 538 nM T70176 C4JKW3 44581167 IC50 = 50 nM T70176 CROB85 44582642 IC50 = 237 nM T70176 C3UIL7 44582684 IC50 = 10600 nM T70176 CN4RC3 44582716 IC50 = 27200 nM T70176 CWHR56 44582744 IC50 = 1160 nM T70176 CZS9G7 44582745 IC50 = 337 nM T70176 COUV96 44582836 IC50 = 149 nM T70176 CL6JO8 44582837 IC50 = 27 nM T70176 C9MG0D 44582838 IC50 = 4090 nM T70176 CD50LG 44587355 IC50 = 44 nM T70176 CYI73P 44587518 IC50 = 875000 nM T70176 C7HG1M 44587519 IC50 = 70000 nM T70176 CPO1C5 44587520 IC50 = 745000 nM T70176 CAO17U 44587538 IC50 = 289000 nM T70176 CD05SO 44587539 IC50 = 91000 nM T70176 CAX04I 44587540 IC50 = 764000 nM T70176 CL71ZV 44587541 IC50 = 816000 nM T70176 CO61WU 44587559 IC50 = 790000 nM T70176 CCNQ05 44587560 IC50 = 1085000 nM T70176 CPU46I 44587561 IC50 = 1002000 nM T70176 CET79F 44587562 IC50 = 1216000 nM T70176 C6HYG9 44587563 IC50 = 262000 nM T70176 C5WQT3 44587603 IC50 = 921000 nM T70176 CAM43E 44587604 IC50 = 926000 nM T70176 C0KDT2 44587605 IC50 = 375000 nM T70176 C79LSO 44587606 IC50 = 417000 nM T70176 CQ49YF 44587676 IC50 = 357000 nM T70176 C3OCZ4 44587677 IC50 = 480000 nM T70176 CJN3G4 44587678 IC50 = 434000 nM T70176 CVJ45H 44587679 IC50 = 386000 nM T70176 C3NO9M 44587680 IC50 = 318000 nM T70176 CWM35B 44587709 IC50 = 611000 nM T70176 CUP9K8 44587710 IC50 = 335000 nM T70176 CHV19Y 44587711 IC50 = 466000 nM T70176 CB6R5Y 44587712 IC50 = 465000 nM T70176 CGY91R 44587713 IC50 = 665000 nM T70176 CFQJ03 44587741 IC50 = 362000 nM T70176 C9U0PO 44587742 IC50 = 1109000 nM T70176 C6H8YK 44587743 IC50 = 438000 nM T70176 CZ9T1N 44587744 IC50 = 296000 nM T70176 CJQ84P 44587745 IC50 = 310000 nM T70176 C4L8CX 44587774 IC50 = 405000 nM T70176 C8NLD0 44587775 IC50 = 340000 nM T70176 CEX7L5 44587776 IC50 = 424000 nM T70176 CH3TD1 44587777 IC50 = 321000 nM T70176 C6PTG1 44587808 IC50 = 92000 nM T70176 CK0MY1 44587809 IC50 = 150000 nM T70176 CK4HG8 44587810 IC50 = 354000 nM T70176 C1OI4M 44587811 IC50 = 312000 nM T70176 C38GTU 44588942 IC50 < 3 nM T70176 C3SO8R 44588964 IC50 = 8 nM T70176 CSQL98 44588989 IC50 = 6 nM T70176 COK2X4 44588990 IC50 = 25 nM T70176 C7IGA8 44588991 IC50 = 400 nM T70176 C2ZVF5 44589014 IC50 = 83 nM T70176 C83PJD 44589040 IC50 = 295 nM T70176 CC5A3R 44589041 IC50 = 23 nM T70176 C7ND9J 44589042 IC50 = 19 nM T70176 CU47KI 44589090 IC50 = 14 nM T70176 CTY03Z 44589091 IC50 = 33 nM T70176 CA5UF3 44589514 Ki > 2500 nM T70176 C3KLD1 44589515 Ki = 1500 nM T70176 C7A0UX 44589516 Ki > 2500 nM T70176 CYK07V 44589517 Ki = 1500 nM T70176 C89COX 44590149 Ki > 5000 nM T70176 C2BQ4M 44590150 Ki = 1652 nM T70176 C6NB9K 44590204 Ki = 1100 nM T70176 CQ0NU8 44590205 Ki = 2400 nM T70176 C4R5DC 44590971 IC50 > 20 ug.mL-1 T70176 CTMD40 44590972 IC50 = 3.8 ug.mL-1 T70176 C36LEO 44590973 IC50 = 4.1 ug.mL-1 T70176 C1PY6R 44590974 IC50 = 3.1 ug.mL-1 T70176 CMH56U 44590975 IC50 = 0.7 ug.mL-1 T70176 CF0LH6 44590976 IC50 = 0.33 ug.mL-1 T70176 C0KTA3 44590977 IC50 = 0.88 ug.mL-1 T70176 CZ5OJ9 44591009 IC50 = 0.55 ug.mL-1 T70176 CC80SY 44591092 IC50 = 2.8 ug.mL-1 T70176 CB8JF4 44591093 IC50 = 0.56 ug.mL-1 T70176 C0QJE3 44591094 IC50 = 12 ug.mL-1 T70176 CG5S0Z 44591095 IC50 = 6.9 ug.mL-1 T70176 C42IQG 44591096 IC50 = 3.6 ug.mL-1 T70176 CX5G9N 44591097 IC50 = 7.1 ug.mL-1 T70176 C28VWN 44591131 IC50 = 1.4 ug.mL-1 T70176 CH7VJ6 44591132 IC50 = 5.5 ug.mL-1 T70176 CH4Y1M 44591133 IC50 = 2.1 ug.mL-1 T70176 C3JVS0 44591386 IC50 = 1.7 ug.mL-1 T70176 CEK87I 44591387 IC50 = 0.35 ug.mL-1 T70176 CAY1Z9 44591388 IC50 = 0.56 ug.mL-1 T70176 CYR7B1 44591389 IC50 = 6.5 ug.mL-1 T70176 CD9G1Q 44591421 IC50 = 12 ug.mL-1 T70176 C57SZQ 44591422 IC50 > 20 ug.mL-1 T70176 C8NL6S 44591423 IC50 > 20 ug.mL-1 T70176 CQ5R0Z 44591424 IC50 > 20 ug.mL-1 T70176 C3FVR5 44591425 IC50 = 8.9 ug.mL-1 T70176 C5Z3LI 44591740 IC50 = 590 nM T70176 C2PX5O 44593468 Ki > 5000 nM T70176 CZ20KC 44593469 Ki > 2500 nM T70176 CM3T7B 44593470 Ki > 2270 nM T70176 CD2FE4 44593471 Ki = 100 nM T70176 CS8GE3 44593472 Ki > 5000 nM T70176 CKM4H0 44593475 Ki > 3330 nM T70176 CV8F0R 44593854 IC50 > 10000 nM T70176 C28QLM 44605035 IC50 > 50000 nM T70176 C75XHS 44605037 IC50 > 50000 nM T70176 C4N3WH 45267635 IC50 = 816000 nM T70176 C2SWY0 45267643 IC50 = 710000 nM T70176 CZHQ40 45267648 IC50 = 960000 nM T70176 CR61WC 45269293 IC50 = 950000 nM T70176 C4W1UX 45269647 IC50 = 81 nM T70176 C7KH5Y 45270972 IC50 = 1210000 nM T70176 CDE0N8 45271900 IC50 = 915000 nM T70176 C9MR8P 45271906 IC50 = 862000 nM T70176 CEIB03 45272690 IC50 = 895000 nM T70176 C74SMH 45272760 IC50 = 1070000 nM T70176 C6OX0V 45375974 IC50 = 410 nM T70176 C6E2SC 45482700 IC50 > 10000 nM T70176 CZXH74 45482750 IC50 > 10000 nM T70176 CX0HO6 45486156 IC50 = 460 nM T70176 CZ58FY 46215814 IC50 = 280 nM T70176 CI1L7W 46222549 IC50 = 0.8 nM T70176 CY3HW5 46224684 IC50 = 140 nM T70176 CM4D1T 46232352 IC50 = 13400 nM T70176 C0JRV8 46232353 IC50 = 18000 nM T70176 CWF4P8 46232354 IC50 > 30000 nM T70176 CA69DW 46232355 IC50 = 5700 nM T70176 CR8SZ3 46232356 IC50 = 16500 nM T70176 C18UZG 46232404 IC50 = 2900 nM T70176 CYT37A 46232443 IC50 > 50000 nM T70176 CF9JK5 46232476 IC50 > 30000 nM T70176 C17VEN 46232477 IC50 > 50000 nM T70176 C3MNW9 46232478 IC50 > 35000 nM T70176 CZS2I3 46232479 IC50 > 35000 nM T70176 C1G3HY 46232521 IC50 > 25000 nM T70176 CTR6C9 46232522 IC50 > 35000 nM T70176 CN8D2T 46232523 IC50 > 35000 nM T70176 CYF51P 46232524 IC50 = 10000 nM T70176 C48ZVW 46232555 IC50 > 50000 nM T70176 CS9B1U 46232556 IC50 > 50000 nM T70176 CC2WT4 46232590 IC50 = 20 nM T70176 CAP27Y 46232738 IC50 > 10000 nM T70176 C5Z0PK 46233015 IC50 > 20000 nM T70176 CYV1U4 46829289 IC50 = 12 nM T70176 CL5K1F 46829290 IC50 = 319 nM T70176 CGO1J5 46830766 Ki = 286 nM T70176 CF7HK2 46830767 Ki = 168 nM T70176 C2HJ1X 46830768 Ki = 522 nM T70176 CLS29B 46872626 IC50 > 10000 nM T70176 CJOM49 46880136 IC50 = 26400 nM T70176 C9WY0Q 46880284 IC50 = 198 nM T70176 C9CKW4 46880292 IC50 = 1070 nM T70176 CROD39 46880293 IC50 = 93 nM T70176 CE1J3N 46880294 IC50 = 117 nM T70176 CE8HO7 46880330 IC50 = 136 nM T70176 CA23RZ 46880364 IC50 = 135 nM T70176 CJT92P 46880365 IC50 = 79 nM T70176 CNQ6Y4 46880366 IC50 = 74 nM T70176 CLQ62J 46880370 IC50 > 2000 nM T70176 CSYB29 46880407 IC50 = 607 nM T70176 CMW01F 46880416 IC50 = 55.3 nM T70176 CW7OT8 46880504 IC50 > 1000 nM T70176 C37GCR 46880505 IC50 > 9000 nM T70176 CJ1B8S 46880932 IC50 = 72 nM T70176 C9TLK1 46880934 IC50 = 104 nM T70176 CQ7ET6 46881853 IC50 = 3160 nM T70176 CDJ57I 46881879 IC50 > 10000 nM T70176 C3T0VS 46911003 IC50 = 500 nM T70176 CFE24L 46911770 IC50 = 1 nM T70176 CP34VL 46929748 IC50 > 1000 nM T70176 CQR9K1 46933384 IC50 > 100000 nM T70176 CWU7F5 49798058 IC50 = 10 nM T70176 CKL1V8 49798556 IC50 > 20000 nM T70176 CBS64G 49830252 IC50 = 13000 nM T70176 CE7D2J 49855568 IC50 = 440 nM T70176 CFD9P3 49855569 IC50 = 440 nM T70176 C1AU5N 49855758 IC50 = 850 nM T70176 CIFK93 49855759 IC50 = 15000 nM T70176 CK48OJ 49855760 IC50 = 2100 nM T70176 CZI3M1 49855761 IC50 = 1900 nM T70176 CRPZ58 49855949 IC50 = 850 nM T70176 CTU0K3 49855950 IC50 = 1200 nM T70176 CF85NL 49855951 IC50 = 1400 nM T70176 CF7YS9 49855952 IC50 = 460 nM T70176 CJU38G 49855953 IC50 = 200 nM T70176 C83VHI 49864785 IC50 > 100000 nM T70176 C2UTK6 49864850 IC50 = 95000 nM T70176 CAE53W 49865153 IC50 > 100000 nM T70176 CNT8C4 49867482 IC50 = 23000 nM T70176 CCL3R5 49867929 IC50 = 900 nM T70176 CAZQ43 51003133 IC50 > 1000 nM T70176 CXA03W 52920796 IC50 > 100 nM T70176 CG85OC 52940761 IC50 = 600 nM T70176 C8BOP9 52942870 IC50 = 5 nM T70176 C0UC1B 52943026 IC50 = 32 nM T70176 C0K5NI 52944208 IC50 = 2200 nM T70176 CY8V0Q 52949108 IC50 = 33 nM T70176 CE8OY2 53317913 IC50 > 100 nM T70176 C2W9OA 53324451 IC50 > 10000 nM T70176 CG50TB 53380598 IC50 = 199.53 nM T70176 CC8G2I 53380599 IC50 = 1584.89 nM T70176 CK52GI 53380818 IC50 = 1100 nM T70176 C1CA4M 53386721 IC50 = 680 nM T70176 CW98EQ 53386722 IC50 > 25000 nM T70176 CJF1M2 53630890 IC50 = 220 nM T70176 CSW32F 54581340 IC50 = 25 nM T70176 C1XS2J 54760383 IC50 > 10000 nM T70176 C9EMO2 54765177 IC50 = 720 nM T70176 CN9QD7 56643097 IC50 = 794.33 nM T70176 C27YEM 56658554 IC50 > 25000 nM T70176 C95GNR 56658555 IC50 > 25000 nM T70176 CX25QL 56658684 IC50 = 9800 nM T70176 CZBP85 56659843 IC50 > 100000 nM T70176 C1ILG0 56659844 IC50 = 10000 nM T70176 C4O1WR 56660107 IC50 = 3162.28 nM T70176 C8G4SB 56662008 IC50 = 190 nM T70176 C49OIA 56662009 IC50 > 25000 nM T70176 CAKY61 56662153 IC50 > 25000 nM T70176 C91IHZ 56663572 IC50 > 15848.93 nM T70176 CQGV57 56665612 IC50 > 25000 nM T70176 CS5XV2 56666509 IC50 = 27000 nM T70176 C4Z2YU 56667019 IC50 = 5011.87 nM T70176 C6U2OQ 56668926 IC50 > 25000 nM T70176 CH72SM 56669073 IC50 > 25000 nM T70176 CC12UJ 56669074 IC50 > 25000 nM T70176 COB07T 56669075 IC50 = 360 nM T70176 C0HA7C 56670167 IC50 = 78 nM T70176 CQ74RS 56670463 IC50 = 12589.25 nM T70176 C7M1CR 56672407 IC50 > 25000 nM T70176 CYJF34 56673688 IC50 = 2700 nM T70176 CR0O6E 56673689 IC50 = 53000 nM T70176 CWV70H 56673950 IC50 = 251.19 nM T70176 C50VCZ 56675790 IC50 > 25000 nM T70176 C4PNF2 56675791 IC50 > 25000 nM T70176 CT3B9L 56675792 IC50 > 25000 nM T70176 CHSX82 56675794 IC50 = 21000 nM T70176 CZMX67 56675913 IC50 > 25000 nM T70176 CQ1OT2 56677279 IC50 = 3981.07 nM T70176 C7ID8C 56677280 IC50 = 5011.87 nM T70176 C9KV5E 56679105 IC50 > 25000 nM T70176 CIK9D5 56679106 IC50 > 25000 nM T70176 CU9IT6 56679107 IC50 > 25000 nM T70176 CQJ9N1 56680334 IC50 = 1100 nM T70176 CU1GX5 56680583 IC50 > 15848.93 nM T70176 COM4F3 56680584 IC50 > 15848.93 nM T70176 CWVS28 56682405 IC50 = 19700 nM T70176 CI7T0B 56682406 IC50 > 25000 nM T70176 CNVL06 56682407 IC50 > 25000 nM T70176 C4OU6L 56682539 IC50 > 25000 nM T70176 CZX9O7 56682540 IC50 > 25000 nM T70176 C2P3RA 56683651 IC50 = 16000 nM T70176 CVLW80 56683909 IC50 = 15848.93 nM T70176 C2MQ6I 56683910 IC50 > 15848.93 nM T70176 CDP30U 56683911 IC50 = 158.49 nM T70176 CA7T5R 56683912 IC50 = 6309.57 nM T70176 CBOD63 56835089 IC50 > 30000 nM T70176 CJBL48 56925034 IC50 = 610 nM T70176 CIV57W 56947168 IC50 = 26600 nM T70176 CR16SD 56947170 IC50 = 4570 nM T70176 CPHX64 57325478 IC50 > 50000 nM T70176 CQ9BW4 57325479 IC50 > 50000 nM T70176 C03XBT 57328467 IC50 > 30000 nM T70176 CXJ35L 57328543 IC50 = 4650 nM T70176 CCF61V 57328544 IC50 = 2020 nM T70176 C39KXI 57328545 IC50 = 6520 nM T70176 CPO2J4 57342178 IC50 = 83 nM T70176 C72PED 57342179 IC50 = 230 nM T70176 CA93PN 57342180 IC50 = 2500 nM T70176 C8X5JG 57384039 IC50 = 26000 nM T70176 CACW05 57386803 IC50 = 2740 nM T70176 CG14VM 57387301 IC50 = 530 nM T70176 CAE9H8 57391299 IC50 > 15848.93 nM T70176 CZ1C4U 57391300 IC50 > 15848.93 nM T70176 C2RV8M 57393078 IC50 > 15848.93 nM T70176 CXA72Y 57393079 IC50 = 5011.87 nM T70176 C16RBI 57393424 IC50 = 4100 nM T70176 CS85QL 57394803 IC50 > 15848.93 nM T70176 C9L2SB 57394812 IC50 = 630.96 nM T70176 CD6Y9Z 57395116 IC50 > 30000 nM T70176 C8W6IG 57395117 IC50 > 30000 nM T70176 CQI0X9 57396562 IC50 = 501.19 nM T70176 CBTP07 57396563 IC50 = 5011.87 nM T70176 CJ6NV4 57396564 IC50 > 15848.93 nM T70176 CK3FP5 57396565 IC50 = 5011.87 nM T70176 CKE3B0 57396576 IC50 = 1995.26 nM T70176 CX17PL 57396577 IC50 = 501.19 nM T70176 CG7S0D 57396882 IC50 > 30000 nM T70176 CE4FA1 57396924 IC50 > 10000 nM T70176 CYR9E5 57398347 IC50 = 501.19 nM T70176 C8B3PI 57398348 IC50 = 630.96 nM T70176 C5CLX0 57400013 IC50 = 3162.28 nM T70176 C0GL5D 57401811 IC50 > 15848.93 nM T70176 C2YZE6 57401822 IC50 = 1258.93 nM T70176 C5OQA0 57403528 IC50 = 3162.28 nM T70176 CHV6R9 57403529 IC50 = 501.19 nM T70176 CLI7S3 57403897 IC50 > 10000 nM T70176 C2GV3D 57523680 Ki = 2000 nM T70176 CBJ6U3 57602135 Ki = 700 nM T70176 C86ICQ 57602171 Ki = 100 nM T70176 CLB9X6 57602200 Ki = 160 nM T70176 CD73BT 57602215 IC50 > 10000 nM T70176 C9NE3U 57602228 IC50 > 10000 nM T70176 CV54XU 57602232 Ki = 2500 nM T70176 CL3WU0 57602368 IC50 > 10000 nM T70176 CKV68E 57602369 Ki = 100 nM T70176 CVK0G4 58056356 IC50 > 50000 nM T70176 C4V7FY 58191950 IC50 = 17000 nM T70176 CPCA29 58191961 IC50 > 100000 nM T70176 C7HF1L 58191965 IC50 = 13000 nM T70176 C8LWY9 58191997 IC50 = 22000 nM T70176 C6BPR2 58985201 IC50 > 50000 nM T70176 CBWJ84 59291203 IC50 = 1030 nM T70176 CZ3TG1 59375154 IC50 = 2700 nM T70176 CXJ63M 59603829 IC50 < 10 nM T70176 CQEU96 59603842 IC50 = 2.2 nM T70176 C16YEO 59662448 IC50 > 50000 nM T70176 COH62U 60097413 IC50 > 3300 nM T70176 C1MR8Q 60097495 IC50 > 5000 nM T70176 C7YPS1 60198399 IC50 = 12 nM T70176 CIG0P8 60198530 IC50 = 9 nM T70176 CR4K5Z 60198532 IC50 = 16 nM T70176 CGT3K9 60198589 IC50 = 23 nM T70176 CK4Z0H 60200097 IC50 = 700 nM T70176 CCON02 60200403 IC50 = 33000 nM T70176 CV8X3M 60200408 IC50 > 100000 nM T70176 CH59YJ 60200737 IC50 = 22000 nM T70176 CCG75S 60200900 IC50 = 62000 nM T70176 CC4V6R 60200902 IC50 = 49000 nM T70176 CG47WK 60200904 IC50 = 21000 nM T70176 CF7M2W 60200906 IC50 = 27000 nM T70176 CN9GQ8 60201066 IC50 = 25000 nM T70176 CRN3D6 60201068 IC50 = 390 nM T70176 C1ER6C 60201070 IC50 = 6400 nM T70176 CR3AJ9 60201072 IC50 > 300000 nM T70176 CR2T5Q 66934034 Ki < 100 nM T70176 C1HSE0 67035086 IC50 = 410 nM T70176 CWI6K5 67035106 IC50 > 10000 nM T70176 C38RGB 67035556 IC50 > 10000 nM T70176 C9WY2P 67383875 Ki = 89 nM T70176 CJY4P6 68212724 IC50 = 114 nM T70176 C8I7GC 68293638 IC50 > 10000 nM T70176 CD56XK 68293660 IC50 > 10000 nM T70176 CNH3R2 68388345 IC50 = 34000 nM T70176 C5L0SQ 68388404 IC50 = 3700 nM T70176 CYI75G 68678653 IC50 > 30000 nM T70176 C5DGR9 69036886 IC50 = 605 nM T70176 CZ4OY5 70681030 IC50 = 345 nM T70176 CPOV92 70681032 IC50 = 155 nM T70176 COHI26 70681033 IC50 = 518 nM T70176 CDB62K 70681398 IC50 > 10000 nM T70176 CN6GK4 70681405 IC50 > 10000 nM T70176 C4TM6F 70682212 IC50 > 30000 nM T70176 C9PE4T 70682214 IC50 > 30000 nM T70176 C7EH1D 70683155 IC50 > 30000 nM T70176 C0NFK3 70683494 IC50 > 10000 nM T70176 CG3C0B 70683495 IC50 > 10000 nM T70176 CDFX37 70683509 IC50 > 10000 nM T70176 CW4C1K 70684312 IC50 > 30000 nM T70176 CRK92N 70685231 IC50 > 5280 nM T70176 CID9O3 70685233 IC50 = 9410 nM T70176 C0WE8F 70685596 IC50 > 10000 nM T70176 CKW18V 70685615 IC50 > 10000 nM T70176 C7OX5Z 70686473 IC50 > 30000 nM T70176 CA0FE8 70687386 IC50 = 135 nM T70176 CQH9A0 70687387 IC50 = 370 nM T70176 CMA7J1 70687388 IC50 = 187 nM T70176 CYHA21 70687748 IC50 > 10000 nM T70176 CEGM27 70689447 IC50 = 70 nM T70176 C80CWD 70689448 IC50 = 2790 nM T70176 C4BSI9 70689798 IC50 > 10000 nM T70176 CN15SY 70691556 IC50 > 4910 nM T70176 CTI38V 70691938 IC50 > 10000 nM T70176 CU07RJ 70691948 IC50 > 10000 nM T70176 CL71AV 70695758 IC50 = 133 nM T70176 C2EI9Z 70695759 IC50 = 1370 nM T70176 CZ4W6K 70695760 IC50 = 3970 nM T70176 CP08FT 70696865 IC50 > 30000 nM T70176 CK58RV 71449587 IC50 = 23 nM T70176 C2HBG8 71450398 IC50 > 50 ug.mL-1 T70176 C6VF7J 71453206 IC50 = 110 nM T70176 C8AH1B 71454033 IC50 > 50 ug.mL-1 T70176 CI37UR 71454035 IC50 > 50 ug.mL-1 T70176 CX3AN8 71454037 IC50 > 50 ug.mL-1 T70176 CO0WF5 71454941 IC50 = 19 nM T70176 CF74SL 71454944 IC50 = 3000 nM T70176 CZG8I6 71456727 IC50 = 16 nM T70176 CE1IX7 71456728 IC50 = 560 nM T70176 C14OGU 71458568 IC50 = 6.7 nM T70176 CVQ62G 71458571 IC50 < 5.2 nM T70176 C74VKX 71458572 IC50 = 31 nM T70176 CM1ND2 71458573 IC50 = 100 nM T70176 C3S0NP 71458574 IC50 = 460 nM T70176 CY6WI2 71458575 IC50 = 7100 nM T70176 C9ZVW4 71459442 IC50 > 50 ug.mL-1 T70176 CO9PR0 71459445 IC50 > 50 ug.mL-1 T70176 C15XAV 71460420 IC50 = 21 nM T70176 CKV1P2 71460421 IC50 = 140 nM T70176 CT7K3A 71460422 IC50 = 520 nM T70176 CB9V6C 71461186 IC50 > 50 ug.mL-1 T70176 C25FQP 71462104 IC50 = 46 nM T70176 C31ZKB 71462893 IC50 = 100 nM T70176 CJ6T0K 71462927 IC50 > 50 ug.mL-1 T70176 CMV23P 71462929 IC50 > 50 ug.mL-1 T70176 CUGP02 71494949 IC50 = 9 nM T70176 CAP8U6 71553522 IC50 > 83000 nM T70176 C53UOG 71560541 IC50 = 8200 nM T70176 CRX81Q 71575642 IC50 > 10000 nM T70176 CQ25SH 71580632 IC50 = 16500 nM T70176 C83CTB 71580633 IC50 = 2700 nM T70176 C5D4KV 71580634 IC50 = 45000 nM T70176 C91YEO 71580635 IC50 = 39000 nM T70176 CYW8T4 71580636 IC50 > 83000 nM T70176 C6BE2H 71580637 IC50 > 29000 nM T70176 CLR9Q7 71580638 IC50 > 83000 nM T70176 CH7C2T 71580737 IC50 > 30600 nM T70176 CEO1Y5 71580738 IC50 = 17000 nM T70176 C92OVF 71580739 IC50 = 5000 nM T70176 CS5DB9 71580740 IC50 = 10000 nM T70176 CI7M6B 71580741 IC50 > 29100 nM T70176 CF14UA 71580742 IC50 = 42000 nM T70176 C5WGV3 71580743 IC50 = 45100 nM T70176 C5JYS4 71580744 IC50 = 3700 nM T70176 CU9LY4 71580745 IC50 = 21000 nM T70176 C4O5VB 71580746 IC50 > 44000 nM T70176 CYZM69 71580828 IC50 = 38000 nM T70176 CN8BT6 71580829 IC50 > 83000 nM T70176 CMS1Y7 71580830 IC50 = 310 nM T70176 CV3K1J 71580831 IC50 = 1100 nM T70176 C9DJ3E 71580832 IC50 = 160 nM T70176 CG32TU 71580833 IC50 = 550 nM T70176 CKZ6E1 71580834 IC50 = 100 nM T70176 CME5Z4 71580835 IC50 = 160 nM T70176 CMAC67 71580913 IC50 = 110 nM T70176 CH54UK 71580914 IC50 > 83000 nM T70176 C6D3HR 71580915 IC50 = 60 nM T70176 C95XJE 71580916 IC50 = 310 nM T70176 C8R9OC 71580917 IC50 > 83000 nM T70176 CBE67N 71731769 IC50 = 3900 nM T70176 CB64IQ 72194525 IC50 = 9.1 nM T70176 C9E4XZ 72546233 IC50 = 580 nM T70176 CE1VB4 72696779 IC50 = 60 nM T70176 CP5AS8 72707650 IC50 = 69 nM T70176 CYG95S 72707651 IC50 = 56 nM T70176 C4U0XJ 72707652 IC50 = 71 nM T70176 C2N1ZE 72707723 IC50 = 52 nM T70176 CNP0V5 72707724 IC50 = 47 nM T70176 CS2E6R 72707725 IC50 = 41 nM T70176 CG5P6E 72707726 IC50 = 63 nM T70176 CY98DU 72707727 IC50 = 42 nM T70176 CU4A5Q 72707728 IC50 = 37 nM T70176 C8Q9PJ 72707787 IC50 = 59 nM T70176 C24YBE 72707788 IC50 = 58 nM T70176 CZ1O6G 72707789 IC50 = 43 nM T70176 CZAM98 72707790 IC50 = 36 nM T70176 CCJ19M 72707791 IC50 = 49 nM T70176 CI3CY4 72707792 IC50 = 44 nM T70176 CQT5S3 72707852 IC50 = 29 nM T70176 CP13FK 72707853 IC50 = 25 nM T70176 CB9K0Z 72707854 IC50 = 32 nM T70176 C75RHB 72707855 IC50 = 30 nM T70176 CBY80T 72716071 IC50 = 4473 nM T70176 CWK32R 72946100 Ki = 2800 nM T70176 CZ57TX 72946278 IC50 > 10000 nM T70176 CHJ9F3 72946279 IC50 > 10000 nM T70176 C79KPC 72946455 IC50 > 10000 nM T70176 C7DQ3G 72946456 IC50 > 10000 nM T70176 CRYA60 72946457 Ki = 2500 nM T70176 CTB12K 72946458 Ki = 300 nM T70176 CNY4H3 73349258 IC50 = 75 nM T70176 C42MXW 76310923 IC50 > 30000 nM T70176 C0MR6F 76310924 IC50 > 30000 nM T70176 C9MG7U 76314564 IC50 > 30000 nM T70176 CU8EW0 76318141 IC50 > 30000 nM T70176 C80VJZ 76318142 IC50 > 30000 nM T70176 C6ZOM5 76321826 IC50 > 30000 nM T70176 C5MRE6 76321827 IC50 = 984 nM T70176 CL0T7B 76322219 IC50 = 18782 nM T70176 C8Z6XR 76325460 IC50 = 13600 nM T70176 CKZ4F9 76325461 IC50 > 30000 nM T70176 CTA86L 76325462 IC50 > 30000 nM T70176 CT1R6E 76329005 IC50 = 1450 nM T70176 CT4FE5 76329006 IC50 > 30000 nM T70176 C7AWU4 76332128 IC50 = 2800 nM T70176 C0PRE8 76336290 IC50 > 30000 nM T70176 CF1JW0 76336291 IC50 > 30000 nM T70176 C7VA5U 78161839 IC50 = 6.4 nM T70176 C2Y1RF 78162193 IC50 < 50 nM T70176 C4NM0V 78162195 IC50 < 50 nM T70176 CWR57U 78357763 IC50 = 96.9 nM T70176 CQ2SU8 78673832 IC50 > 30000 nM T70176 CE0W9R 78673833 IC50 > 30000 nM T70176 CV8UZ1 86278565 IC50 = 93 nM T70176 C8VP5N 86298673 IC50 = 10 nM T70176 CPG3A5 86302574 IC50 > 30000 nM T70176 CA49FO 86705475 IC50 = 11 nM T70176 C1HW4B 89735655 IC50 = 51 nM T70176 CV64KY 90183363 IC50 = 2220 nM T70176 CL4JO2 90183809 IC50 = 80 nM T70176 CXV2R0 90645247 IC50 = 2 nM T70176 C90SKQ 90645248 IC50 = 2 nM T70176 CXZ0H7 90645249 IC50 = 104 nM T70176 C1Z6GR 90645250 IC50 = 13 nM T70176 C3CGL5 90645251 IC50 = 821 nM T70176 C8BPR2 90645252 IC50 = 71 nM T70176 C8FOU6 90645255 IC50 = 69 nM T70176 CDWB05 90645256 IC50 = 13 nM T70176 CWE9I2 91664021 IC50 > 10000 nM T70176 CW58AE 91664022 IC50 > 10000 nM T70176 CB25UZ 91664023 IC50 > 10000 nM T70176 C8W9KV 91844733 IC50 = 620 nM T70176 CAU45T 91971978 IC50 > 30000 nM T70176 CRI0S4 101891768 IC50 = 530 nM T70176 CL64EZ 102287891 IC50 > 10000 nM T70176 C2NQ4S 102287892 IC50 > 10000 nM T70176 CZG9I3 118030039 IC50 = 4 nM T70176 CX58DI 118716791 IC50 > 30000 nM T70176 CD9X2B 118716796 IC50 > 30000 nM T70176 C2YJ0O 118716797 IC50 > 30000 nM T70176 CL3UO9 118716798 IC50 > 30000 nM T70176 C71BAM 118716799 IC50 > 30000 nM T70176 CU4EL6 118716806 IC50 > 30000 nM T70176 CI5W9H 118720010 IC50 = 503 nM T70176 COQ9S4 118720011 IC50 = 476 nM T70176 CHT6K9 118728811 Ki > 4000 nM T70176 CUA3Y2 118728812 Ki > 4000 nM T70176 CDQ78G 118728813 Ki > 4000 nM T70176 CZ6XL7 118728814 Ki > 4000 nM T70176 CMO67K 118728815 Ki > 4000 nM T70176 CR2M0Q 118728816 Ki > 4000 nM T70176 C62SCL 118728817 Ki > 4000 nM T70176 CSB30C 118728819 Ki > 4000 nM T70176 CV7XU8 118728820 Ki > 4000 nM T70176 C3J1EX 118728821 Ki > 4000 nM T70176 CIWB78 118728822 Ki > 4000 nM T70176 CP18SE 118728823 Ki = 1200 nM T70176 CM42CA 118728824 Ki > 4000 nM T70176 C9Q7CL 118728825 Ki > 4000 nM T70176 CCR3S0 118728826 Ki > 4000 nM T70176 CP27TX 118735321 IC50 = 33215 nM T70176 CJH0M1 118735322 IC50 = 577 nM T70176 CA7Z4X 118735323 IC50 = 12295 nM T70176 C76XKT 118735324 IC50 = 14060 nM T70176 CI26FD 118735325 IC50 = 14789 nM T70176 CU8T1C 118735326 IC50 = 1995 nM T70176 C1PDE5 118735327 IC50 = 1819 nM T70176 CQ0GS4 118735328 IC50 = 10476 nM T70176 C3KLT1 118735329 IC50 = 17368 nM T70176 C1RAP6 118735330 IC50 = 13713 nM T70176 CQ45PF 118735331 IC50 = 20 nM T70176 C56MYE 118735332 IC50 = 45885 nM T70176 CP26VF 118735333 IC50 = 16884 nM T70176 CSR3N8 118735334 IC50 > 100000 nM T70176 C3TS7H 118735335 IC50 > 100000 nM T70176 C4DQ5K 118735336 IC50 = 5176 nM T70176 C4DQX9 118735337 IC50 = 38379 nM T70176 CBY4K3 118735338 IC50 = 56703 nM T70176 C5CK7W 118735339 IC50 = 314 nM T70176 CQCX41 118737057 IC50 > 10000 nM T70176 CV06MA 122177111 IC50 = 392 nM T70176 C2DH7M 122177112 IC50 = 392 nM T70176 C8GB4Q 122181008 IC50 > 10000 nM T70176 CBQ94Z 122181009 IC50 > 10000 nM T70176 CT8CP2 122181010 IC50 > 10000 nM T70176 CB6IZ0 122181011 IC50 > 10000 nM T70176 C65BOF 122181012 IC50 > 10000 nM T70176 CO83PN 122181013 IC50 > 10000 nM T70176 C69ULZ 122181014 IC50 > 100000 nM T70176 CN14DV 122181015 IC50 > 10000 nM T70176 CIG8Y1 122181016 IC50 > 10000 nM T70176 CRJS41 122181017 IC50 > 10000 nM T70176 CVB03H 122181018 IC50 > 10000 nM T70176 C6SJ3X 122181019 IC50 > 10000 nM T70176 C58CJI 122181022 IC50 > 10000 nM T70176 CG2Z8B 122181023 IC50 > 10000 nM T70176 CC2G8N 122181024 IC50 > 10000 nM T70176 CM2DU7 122181025 IC50 > 10000 nM T70176 C5YB3O 122181096 IC50 > 10000 nM T70176 CV5BQ9 122181097 IC50 > 10000 nM T70176 CFKD32 122191637 IC50 > 50000 nM T70176 C4X7SD 122192466 IC50 > 10000 nM T70176 COF75Z 126970673 IC50 = 700 nM T70176 C4PFZ0 127046319 IC50 = 5700 nM T70176 C0CX4P 127046320 IC50 = 4000 nM T70176 CUD8G5 127046367 IC50 = 11000 nM T70176 CA83YU 127047442 IC50 = 1400 nM T70176 CNJQ71 127047443 IC50 = 3400 nM T70176 CC1VO7 127047444 IC50 > 25000 nM T70176 CS6C8O 127050851 IC50 = 1520 nM T70176 C1HAU4 127050852 IC50 = 1380 nM T70176 CHVU86 127050853 IC50 = 545 nM T70176 CWDX26 127050854 IC50 = 113 nM T70176 C7DU0N 127050855 IC50 = 832 nM T70176 CDJQ32 127051599 IC50 = 25 nM T70176 C2ISZ9 127051600 IC50 = 494 nM T70176 C61GFX 127051601 IC50 = 135 nM T70176 CFQ2X7 127051618 IC50 = 232 nM T70176 C4DSF7 127051619 IC50 = 1680 nM T70176 C8JMN0 127051620 IC50 = 361 nM T70176 CTZK49 127051621 IC50 = 63 nM T70176 C7PZM3 127051622 IC50 = 254 nM T70176 C4Q5LF 132471857 IC50 = 3800 nM T70176 CJ3M5I 134137436 Ki > 1000 nM T70176 C1MTG5 134543905 IC50 > 200 nM T70176 CLSE63 135398512 IC50 = 1330 nM T70176 CS4OW8 135400873 Ki = 340 nM T70176 COYA04 135402863 IC50 = 50 nM T70176 C4OWM1 135403014 IC50 = 9 nM T70176 C9Y3WG 135404113 IC50 = 17 nM T70176 CDV48Y 135404796 IC50 = 13 nM T70176 CUY41E 135404846 IC50 = 1 nM T70176 CFOD89 135405216 IC50 = 10 nM T70176 CF39KX 135405229 IC50 = 28 nM T70176 CS7QH2 135405282 IC50 = 2.1 nM T70176 C82TVC 135409809 IC50 = 1.5 nM T70176 C8S0OH 135416016 IC50 = 5 nM T70176 C3YPB0 135416046 IC50 = 60 nM T70176 CH98WL 135418427 IC50 = 54 nM T70176 CL46JK 135418490 IC50 = 2.3 nM T70176 C5ZQ0M 135421134 IC50 = 360 nM T70176 CE8LA2 135421135 IC50 = 22 nM T70176 CWO64E 135421136 IC50 = 2.5 nM T70176 C3U0PF 135421137 IC50 = 2 nM T70176 C3A9UZ 135421138 IC50 = 8.9 nM T70176 C30VGC 135421139 IC50 = 310 nM T70176 CRA56X 135421140 IC50 = 2.1 nM T70176 CT0D5M 135421141 IC50 = 3 nM T70176 CXZV53 135421142 IC50 = 1.9 nM T70176 CTRW73 135421143 IC50 = 61 nM T70176 CC84WV 135421144 IC50 = 2.8 nM T70176 C7TW3I 135421145 IC50 = 1.5 nM T70176 C9DUQ7 135421146 IC50 = 5.6 nM T70176 C3ERJ8 135421147 IC50 = 4.6 nM T70176 C13RGY 135421148 IC50 = 4.7 nM T70176 CEQ2X6 135421149 IC50 = 3.6 nM T70176 CE7LR5 135421150 IC50 = 0.54 nM T70176 C07BWX 135421151 IC50 = 4.5 nM T70176 CBUN39 135421152 IC50 = 4.3 nM T70176 CID92J 135421153 IC50 = 5.6 nM T70176 C29QXJ 135421154 IC50 = 281 nM T70176 CFB7R0 135421155 IC50 = 5.6 nM T70176 CK7Y5X 135421156 IC50 = 75 nM T70176 C3R8LM 135421157 IC50 = 1000 nM T70176 C4SIP0 135421158 IC50 = 5.7 nM T70176 CMN0Q7 135421159 IC50 = 7.5 nM T70176 C6J9YR 135421160 IC50 = 26 nM T70176 CH50XP 135421161 IC50 = 50 nM T70176 CY53SU 135421162 IC50 = 14 nM T70176 C3S7MX 135423008 IC50 > 1000 nM T70176 CYG2V6 135428039 IC50 = 160 nM T70176 C4CXD1 135434964 IC50 = 120 nM T70176 CFK9A4 135434965 IC50 = 30 nM T70176 C0ETV8 135434966 IC50 = 4.6 nM T70176 C9VM6D 135434967 IC50 = 7.9 nM T70176 CYBG82 135434968 IC50 = 2.5 nM T70176 C14BLP 135434969 IC50 = 1.2 nM T70176 CX16AQ 135434970 IC50 = 93 nM T70176 C3EU9C 135434971 IC50 = 3.4 nM T70176 C86TJA 135434972 IC50 = 13 nM T70176 C1QYE8 135434973 IC50 = 21 nM T70176 CZ63UC 135434975 IC50 = 12 nM T70176 CP95VZ 135434976 IC50 = 19 nM T70176 C52GQD 135434977 IC50 = 2400 nM T70176 C34YNR 135434978 IC50 = 34 nM T70176 CSLE24 135434979 IC50 = 11 nM T70176 CQT79I 135434980 IC50 = 12 nM T70176 CLP2K4 135434981 IC50 = 15 nM T70176 C8ZS4W 135434982 IC50 = 74 nM T70176 C9XT7W 135434983 IC50 = 16 nM T70176 C6I1SH 135434984 IC50 = 43 nM T70176 C3S7WD 135434985 IC50 = 15 nM T70176 C45SHY 135434986 IC50 = 4.5 nM T70176 CSZ68Y 135434987 IC50 = 12 nM T70176 CN4MJ6 135434988 IC50 = 25 nM T70176 C2C3RF 135434989 IC50 = 8.9 nM T70176 CLYV03 135434990 IC50 = 6.8 nM T70176 CP8GA6 135434991 IC50 = 1.7 nM T70176 CN3A8I 135434992 IC50 = 43 nM T70176 CCP04J 135434993 IC50 = 21 nM T70176 C2VI7F 135434994 IC50 = 75 nM T70176 CBV6K4 135434995 IC50 > 1000 nM T70176 CY8W1P 135434996 IC50 > 1000 nM T70176 C1TN2K 135435000 IC50 = 13 nM T70176 CDM9R4 135435001 IC50 = 54 nM T70176 C7M6WJ 135435002 IC50 = 4.6 nM T70176 CZSD45 135435003 IC50 = 13 nM T70176 CL0YS2 135435004 IC50 = 2.2 nM T70176 C64JZD 135435005 IC50 = 9.5 nM T70176 CGD0F2 135435006 IC50 = 7.1 nM T70176 CH41JZ 135435007 IC50 = 1.6 nM T70176 C52RQG 135435008 IC50 = 13 nM T70176 CPFI68 135435011 IC50 = 5 nM T70176 CS14KX 135435016 IC50 = 2 nM T70176 C2ICP3 135435017 IC50 = 2 nM T70176 C6AZ2R 135435018 IC50 = 5 nM T70176 CBUR78 135435019 IC50 = 12.6 nM T70176 CEK04O 135436430 IC50 = 37000 nM T70176 CRI23H 135436431 IC50 = 24000 nM T70176 CM4J6A 135444580 IC50 = 88 nM T70176 C8GZ2B 135449326 Ki > 4000 nM T70176 CCU3G9 135450829 IC50 = 3.3 nM T70176 C8PRH9 135516527 IC50 = 21 nM T70176 CTJ48K 135524085 IC50 = 8200 nM T70176 CUT1W7 135524168 IC50 > 10000 nM T70176 CTB7R2 135564980 IC50 = 15000 nM T70176 C6QA2T 135566358 IC50 = 530 nM T70176 CJN0Z7 135566360 IC50 = 1800 nM T70176 CZY5G2 135566361 IC50 = 52 nM T70176 C7ER0S 135566450 IC50 = 10000 nM T70176 CUC08B 135566451 IC50 = 1040 nM T70176 CY4D8I 135566504 Ki > 1000 nM T70176 CM6C9G 135566570 IC50 = 68 nM T70176 C7PJ6X 135566704 IC50 > 30000 nM T70176 CFAD48 135611170 Ki > 2000 nM T70176 CPV59N 135685787 Ki = 62 nM T70176 C95JVR 135744117 IC50 = 9.3 nM T70176 C6Q8IN 135839312 IC50 = 102 nM T70176 C2SE7D 135863109 IC50 = 8400 nM T70176 CX4ZB3 135863110 IC50 = 4700 nM T70176 C6B4OS 135863111 IC50 > 50000 nM T70176 CC63MW 135863112 IC50 > 50000 nM T70176 CST7X3 135870706 IC50 < 50 nM T70176 CV24UR 135873213 IC50 = 2 nM T70176 C8P2FB 135875593 IC50 = 2600 nM T70176 CN0S3W 135875595 IC50 = 12500 nM T70176 CAP19T 135875596 IC50 = 17300 nM T70176 CZ4RQ6 135875597 IC50 = 16900 nM T70176 C01DTS 135875598 IC50 = 6900 nM T70176 COU3P4 135875600 IC50 = 6600 nM T70176 CD8U9R 135875601 IC50 < 50000 nM T70176 CSOR81 135875602 IC50 = 3100 nM T70176 C2BI9W 135875603 IC50 < 50000 nM T70176 C49XYF 135875604 IC50 = 870 nM T70176 CKJ85A 135875605 IC50 = 2900 nM T70176 CF4GP1 135875606 IC50 = 3100 nM T70176 CDP2N8 135875607 IC50 = 18300 nM T70176 CYNW03 135875608 IC50 = 1100 nM T70176 C4MYH7 135875609 IC50 < 25900 nM T70176 CDUV39 135875610 IC50 < 50000 nM T70176 C1EXP2 135875611 IC50 < 34500 nM T70176 CWSN64 135875612 IC50 < 50000 nM T70176 CP9BQ0 135875613 IC50 < 50000 nM T70176 CXR7C9 135875614 IC50 = 6700 nM T70176 CK3FH5 135875615 IC50 = 6100 nM T70176 CN4E9Q 135875616 IC50 < 50000 nM T70176 CTGF14 135875617 IC50 = 45500 nM T70176 C6UP5Q 135875618 IC50 = 15100 nM T70176 C36TXV 135875619 IC50 = 3600 nM T70176 CAHI68 135875620 IC50 = 2700 nM T70176 CG8X9Z 135875621 IC50 = 13600 nM T70176 C12XZF 135875622 IC50 = 2600 nM T70176 CH8RT2 135875623 IC50 = 16900 nM T70176 CTL0R1 135875624 IC50 = 41500 nM T70176 C9S7CR 135875716 IC50 > 50000 nM T70176 C4U1XR 135875719 IC50 > 50000 nM T70176 CN4CX8 135875746 IC50 > 50000 nM T70176 CF0CM3 135909510 IC50 = 990 nM T70176 CVH9A7 135909511 IC50 = 140 nM T70176 CWIE69 135909512 IC50 = 230 nM T70176 CGSC82 135909513 IC50 = 1200 nM T70176 CQ1RH0 135909514 IC50 = 160 nM T70176 CLVK24 135922684 IC50 = 960 nM T70176 CF6N2M 135922716 IC50 = 1600 nM T70176 C8Z7VH 135922717 IC50 = 2600 nM T70176 C79ZPW 135922718 IC50 = 2300 nM T70176 CV1O5B 135922720 IC50 = 1300 nM T70176 C1C3XE 135922728 IC50 = 500 nM T70176 CBRZ35 135922729 IC50 = 1200 nM T70176 C70SDW 135922730 IC50 = 1900 nM T70176 CPJ06A 135922731 IC50 > 50000 nM T70176 CR8K2O 135922732 IC50 = 700 nM T70176 CG3UZ1 135927974 Ki > 1000 nM T70176 COM64Y 135928471 IC50 = 4.1 nM T70176 CYV4X9 135928472 IC50 = 13.3 nM T70176 C7N0LZ 135928473 IC50 = 21500 nM T70176 CN0CT1 135928474 IC50 = 10000 nM T70176 CF94AE 135928475 IC50 = 10000 nM T70176 CN28FB 135928476 IC50 = 10000 nM T70176 CDO4A0 135928477 IC50 = 6100 nM T70176 CG0JQ5 135928478 IC50 = 1730 nM T70176 CHX3L1 135928479 IC50 = 247 nM T70176 C1P9EO 135928480 IC50 = 10000 nM T70176 CIR82V 135928481 IC50 = 10000 nM T70176 CE2K9B 135928482 IC50 = 109000 nM T70176 CR0M6N 135928484 IC50 = 10000 nM T70176 C4POF5 135928485 IC50 = 10000 nM T70176 CQK06T 135928488 IC50 = 10000 nM T70176 CGC14V 135930678 IC50 = 24000 nM T70176 CF1PS8 135934877 Ki = 95 nM T70176 C4QI5M 135939768 IC50 > 50000 nM T70176 CF3GL7 135939769 IC50 > 50000 nM T70176 CR48QX 135939770 IC50 > 50000 nM T70176 CN2A1B 135939771 IC50 > 50000 nM T70176 CKGI27 135939772 IC50 > 50000 nM T70176 CFPI38 135939773 IC50 > 50000 nM T70176 CQW25F 135939775 IC50 > 50000 nM T70176 CG09ML 135939776 IC50 = 20400 nM T70176 C5F6YN 135939777 IC50 = 8100 nM T70176 CBKW84 135939778 IC50 > 50000 nM T70176 CZ0F5J 135939779 IC50 > 50000 nM T70176 CN39WJ 135939780 IC50 > 50000 nM T70176 CUX4M6 135939781 IC50 > 50000 nM T70176 CNAL21 135939782 IC50 > 50000 nM T70176 CE6QC1 135939783 IC50 > 50000 nM T70176 CE3PW5 135939784 IC50 > 50000 nM T70176 CXB4R0 135939785 IC50 = 26500 nM T70176 CA8M2E 135939786 IC50 > 50000 nM T70176 CXT6Y3 135939788 IC50 > 50000 nM T70176 C19DFT 135939802 IC50 > 28000 nM T70176 CWNS19 135939803 IC50 > 29000 nM T70176 CJF15Y 135939804 IC50 = 21000 nM T70176 C6LR8O 135939805 IC50 = 19600 nM T70176 CP5R0X 135939806 IC50 = 47000 nM T70176 C2M5XR 135939807 IC50 > 50000 nM T70176 CT8P5L 135939811 IC50 > 50000 nM T70176 CHEQ58 135939812 IC50 = 47000 nM T70176 CE19UY 135939813 IC50 > 50000 nM T70176 C2UN4G 135939814 IC50 > 50000 nM T70176 CN14EI 135939815 IC50 > 50000 nM T70176 CDG7S6 135939816 IC50 = 39800 nM T70176 C5EL7X 135939817 IC50 > 50000 nM T70176 C5Z8HM 135939818 IC50 > 50000 nM T70176 CTH80P 135939819 IC50 > 50000 nM T70176 C41UKD 135939820 IC50 > 50000 nM T70176 COF12L 135939821 IC50 > 50000 nM T70176 C03AVC 135939822 IC50 > 50000 nM T70176 CNE35S 135939823 IC50 = 7700 nM T70176 CS0CH7 135939825 IC50 > 50000 nM T70176 C7MQR3 135939826 IC50 > 50000 nM T70176 COJ3I9 135939827 IC50 > 50000 nM T70176 C9AUC5 135939828 IC50 > 50000 nM T70176 CA89CK 135939829 IC50 > 50000 nM T70176 CGP23U 135939830 IC50 > 50000 nM T70176 CZ4V1F 135939831 IC50 > 50000 nM T70176 CXP61U 135939833 IC50 > 50000 nM T70176 CVF49U 135939834 IC50 > 50000 nM T70176 CMNJ39 135939835 IC50 > 50000 nM T70176 CJ34DP 135939836 IC50 > 50000 nM T70176 CTRL59 135976660 Ki = 76 nM T70176 C97HEY 136007770 IC50 = 50 nM T70176 C8BLU3 136007771 IC50 = 42 nM T70176 C3GVB5 136007772 IC50 = 90 nM T70176 C5NBU3 136025846 IC50 = 450 nM T70176 CEPW57 136025847 IC50 = 60 nM T70176 CT0N5U 136025985 IC50 > 10000 nM T70176 CFNZ81 136025987 IC50 = 2110 nM T70176 CJPT24 136025988 IC50 = 42 nM T70176 CWD1J4 136025989 IC50 = 250 nM T70176 CL1NP0 136026131 IC50 = 21 nM T70176 C9P4LG 136026476 IC50 > 10000 nM T70176 C1PCJ3 136042251 IC50 = 7000 nM T70176 CU56DT 136045789 IC50 > 50000 nM T70176 CA0JB4 136068686 IC50 > 10000 nM T70176 C5BGL2 136068687 IC50 = 360 nM T70176 CXK3F8 136086909 IC50 = 15 nM T70176 CBC27R 136086910 IC50 = 52 nM T70176 CSM28V 136086911 IC50 = 200 nM T70176 C7FU8S 136086912 IC50 = 450 nM T70176 CWH74C 136086913 IC50 = 300 nM T70176 C60YSD 136086914 IC50 = 790 nM T70176 CXV64Q 136086915 IC50 = 940 nM T70176 C59GAN 136086916 IC50 = 3760 nM T70176 C20UHS 136086917 IC50 = 3980 nM T70176 C3X8QG 136086918 IC50 > 10000 nM T70176 C9KV0Y 136086919 IC50 > 10000 nM T70176 CM5T4K 136176135 Ki = 3.4 nM T70176 CQ84IZ 136180335 Ki > 4000 nM T70176 CZ7EX0 136183413 IC50 = 4000 nM T70176 CXFM96 136184114 IC50 = 10000 nM T70176 C72FRE 136184116 IC50 = 5 nM T70176 CRO6H1 136203706 IC50 = 4500 nM T70176 CY36QB 136254272 IC50 = 14000 nM T70176 C61DOF 136274355 IC50 = 9.5 nM T70176 C0EV4N 136845708 IC50 > 91000 nM T70176 CH3M4B 137083628 IC50 > 30000 nM T70176 CJA07O 137083629 IC50 > 30000 nM T70176 C9F8PX 137083630 IC50 > 30000 nM T70176 CNFE23 137349058 IC50 = 120 nM T70176 CV6KR8 137349062 IC50 = 180 nM T70176 C8DF0S 137349068 IC50 = 610 nM T70176 C7Y1KN 137349069 IC50 = 47000 nM T70176 CURM83 137349070 IC50 = 30 nM T70176 CW91ZR 137628992 IC50 = 150000 nM T70176 CMS41L 137628993 IC50 = 9300 nM T70176 CM26KA 137628998 IC50 = 570 nM T70176 CJ2QX1 137629178 IC50 = 2900 nM T70176 CMY9I7 137629183 IC50 = 19000 nM T70176 CBDU81 137629200 IC50 = 570 nM T70176 CI1E8V 137634241 IC50 > 10000 nM T70176 C8GQD5 137636872 IC50 = 370 nM T70176 C7TG3J 137641313 IC50 = 1000 nM T70176 C3W4RO 138403252 IC50 = 37000 nM T70176 CB98HD 145950262 IC50 = 25.4 nM T70176 C7PU6X 145956666 IC50 = 21.5 nM T70176 CK81WV 145957463 IC50 = 190 nM T70176 CJ4FO8 145957807 IC50 = 81.54 nM T70176 CDNC31 145967951 IC50 > 500 nM T70176 CXS4L8 145975683 IC50 = 6700 nM T70176 CB2J4N 145989210 IC50 = 1 nM T70176 CR2GW6 145994117 IC50 = 90 nM T70176 C42TMN 155523743 IC50 = 57 nM T70176 C6RB5J 155534811 IC50 = 630 nM T70176 C8OC5N 155537111 IC50 > 200 nM T70176 CK3EW2 155545512 IC50 = 580 nM T70176 CZQM57 155554194 IC50 > 10000 nM T70176 CETH36 155557337 IC50 > 200 nM T70176 CLXN40 155565350 IC50 = 5 nM T70176 C70ZUA 155569262 IC50 = 1270 nM T70176 D00ERW 44444843 Ki = 3088 nM T70176 D00HVA 11624601 Ki = 820 nM T70176 D00MXS 5281703 IC50 = 1460 nM T70176 D01LPG 9994066 IC50 = 1900 nM T70176 D01MNK 25125014 IC50 = 3 nM T70176 D02DLC 6539361 IC50 = 1.995 nM T70176 D03BJF 44465558 IC50 = 630 nM T70176 D03DZO 11715767 IC50 = 240 nM T70176 D03VDM 787236 IC50 = 855000 nM T70176 D04NGS 5330790 IC50 = 2 nM T70176 D04PEI 11467730 IC50 = 29000 nM T70176 D04RBG 3536 IC50 = 9.7 nM T70176 D04TLB 135408762 IC50 = 9 nM T70176 D04TPA 72163809 IC50 = 7200 nM T70176 D04WFN 10202471 IC50 = 400 nM T70176 D04YQF 763936 IC50 = 25000 nM T70176 D06HVH 54613583 IC50 > 10000 nM T70176 D06LJL 9916282 IC50 = 62000 nM T70176 D06QWO 14824655 IC50 > 10 ug.mL-1 T70176 D07ADR 2422 IC50 = 800 nM T70176 D07ADX 54764565 IC50 = 1180 nM T70176 D07HPE 481747 IC50 > 200000 nM T70176 D07OAT 456214 IC50 = 70 nM T70176 D07ODE 680935 IC50 = 97000 nM T70176 D07SGT 87031 IC50 = 120000 nM T70176 D08RZB 11153014 IC50 > 25000 nM T70176 D09OAH 73292 IC50 = 500000 nM T70176 D0C7RS 1369 IC50 = 91000 nM T70176 D0CM6T 11314340 Ki = 46 nM T70176 D0D3HB 9926933 IC50 = 660 nM T70176 D0G2CT 3708 IC50 = 22 nM T70176 D0G3SZ 6918469 IC50 > 10 ug.mL-1 T70176 D0GT8N 5154691 IC50 = 5 nM T70176 D0H3EV 5005498 IC50 = 15 nM T70176 D0I1FJ 11393719 IC50 > 10000 nM T70176 D0IR6U 5494425 IC50 = 3300 nM T70176 D0J3LR 11634725 Ki = 852 nM T70176 D0KH5T 5687 IC50 = 1000 nM T70176 D0L0HG 766949 IC50 > 10000 nM T70176 D0L3FK 5289419 IC50 = 22 nM T70176 D0M5PI 10730551 IC50 = 4500 nM T70176 D0ME9B 46868971 IC50 > 10 nM T70176 D0MF5Y 5281614 IC50 = 5000 nM T70176 D0MK6D 449088 IC50 = 289.73 nM T70176 D0O0VP 6539367 Ki = 50 nM T70176 D0P6JS 11675054 IC50 < 1 nM T70176 D0Q0YV 24944925 IC50 = 154.88 nM T70176 D0Q3NG 11715520 Ki > 8600 nM T70176 D0QI7H 1540 IC50 = 2300 nM T70176 D0R1FT 4564 Ki = 1200 nM T70176 D0S7IE 11658882 Ki = 1300 nM T70176 D0T4SJ 10356352 IC50 = 140 nM T70176 D0T8NU 16757525 IC50 = 138 nM T70176 D0U0GE 447956 Ki = 396 nM T70176 D0U8YN 398148 Ki = 1300 nM T70176 D0W0PF 118458 IC50 = 350000 nM T70176 D0W7TU 947057 IC50 > 50000 nM T70176 D0X5LN 688798 IC50 > 500000 nM T70176 D0Y5RO 4566 IC50 = 5 nM T70176 D0Y6DX 447649 IC50 = 1000 nM T70176 D0YM4A 22319604 IC50 = 2500 nM T70176 D0YZ7H 9797370 IC50 > 10000 nM T72444 D0YV1Q 6032 IC50 = 6800 nM T72444 C7S5BZ 71525152 IC50 = 1600 nM T72444 CY2V9M 91810296 IC50 = 6200 nM T72444 C96VED 118721937 IC50 = 5200 nM T72444 CQV23Z 118721938 IC50 = 6100 nM T72444 C7NUT9 118721939 IC50 = 7200 nM T72444 C6QA4B 118721940 IC50 = 4900 nM T72444 COF6J8 118721941 IC50 = 8600 nM T72444 CW41SN 118721942 IC50 = 9200 nM T72444 CQKP40 118721943 IC50 = 20800 nM T72444 CT7LE9 118721944 IC50 = 13500 nM T72444 C1BEO7 118722297 IC50 = 36200 nM T72444 C3G0TE 137631437 IC50 = 3500 nM T72444 C5Z4HF 137631862 IC50 = 3900 nM T72444 CTK1D7 137633529 IC50 = 8900 nM T72444 CZ6I1M 137633813 IC50 = 24100 nM T72444 C4DV5G 137635459 IC50 = 12400 nM T72444 C1AOS2 137639300 IC50 = 5100 nM T72444 CU01XC 137640399 IC50 = 6900 nM T72444 CE8MU9 137640444 IC50 = 6700 nM T72444 CV1U7M 137640872 IC50 = 3900 nM T72444 CLGP26 137641910 IC50 = 17600 nM T72444 C62OGI 137643704 IC50 = 4100 nM T72444 CX4PJ0 137644811 IC50 = 7800 nM T72444 CFGU74 137645062 IC50 = 9500 nM T72444 CZN0W4 137648783 IC50 = 38700 nM T72444 CC71JR 137648958 IC50 = 4300 nM T72444 CGV01O 137650837 IC50 = 5200 nM T72444 CGY94A 137652877 IC50 = 5400 nM T72444 CB4JF8 137654288 IC50 = 13200 nM T72444 CC59UQ 137657672 IC50 = 4700 nM T72444 CHS19T 137657734 IC50 = 4600 nM T72444 C9QG2F 137658087 IC50 = 20600 nM T72444 CC8PT3 137659121 IC50 = 2000 nM T72444 C3I9YC 137660475 IC50 = 4400 nM T72444 CU7P9L 137660970 IC50 = 7200 nM T72444 CO39ZV 137661831 IC50 = 32500 nM T72444 D0M5WG 439318 IC50 = 5600 nM T07303 D01PZD 5329098 IC50 = 50 nM T07303 D01ZRI 6450551 IC50 = 0.1 nM T07303 D0G6QF 3081361 IC50 = 233 nM T07303 D0IQ6P 25102847 IC50 = 6 nM T07303 D0R0FO 9823820 IC50 = 5.2 nM T07303 D0R0MW 5329102 IC50 = 8.9 nM T07303 D0W5HK 216239 IC50 = 3 nM T07303 D00DRL 44137946 IC50 = 78 nM T07303 D02RJY 11442891 IC50 = 161 nM T07303 D02WVT 25031915 IC50 = 10 nM T07303 D03HUX 49792852 IC50 > 10000 nM T07303 D03LWG 53235510 IC50 = 2072 nM T07303 D03QLG 9917013 IC50 = 39 nM T07303 D05EXN 58298316 IC50 = 651 nM T07303 D05PZB 135398495 IC50 = 1 nM T07303 D06DMQ 59472121 Ki = 8 nM T07303 D07HRU 9549295 IC50 = 125 nM T07303 D07KYT 24889392 IC50 = 4900 nM T07303 D07NOI 9808844 IC50 = 4 nM T07303 D09VMI 9933475 IC50 = 3 nM T07303 D0D1GF 42642645 IC50 = 2.8 nM T07303 D0E3TC 44259 IC50 = 0.9 nM T07303 D0H9FR 118295624 IC50 = 410 nM T07303 D0IQ0Z 46885626 IC50 = 74 nM T07303 D0M0XB 10302451 IC50 > 10000 nM T07303 D0M9QZ 11485656 IC50 = 12.59 nM T07303 D0O0LS 25141092 IC50 > 1000 nM T07303 D0P1CV 46191454 IC50 > 10000 nM T07303 D0P6DJ 151194 IC50 = 195 nM T07303 D0Q9UX 16718576 IC50 = 920 nM T07303 D0SG7B 49831257 IC50 = 274 nM T07303 D0T2ER 24767976 IC50 = 1.1 nM T07303 D0W7JZ 9911830 IC50 = 0.24 nM T07303 D00DQX 11667893 IC50 = 6 nM T07303 D0H4GI 10275001 IC50 = 4 nM T07303 D0T3ME 156422 IC50 = 270 nM T07303 C63WLY 89644 IC50 = 9.9 ug.mL-1 T07303 CE4K5D 92516 IC50 > 50000 nM T07303 C5JE2Z 104860 IC50 = 2.8 ug.mL-1 T07303 C6Y9CV 151193 IC50 = 195 nM T07303 CI1NA5 159926 IC50 > 10 ug.mL-1 T07303 CI80NA 160436 IC50 > 50000 nM T07303 CYBA43 177458 IC50 = 2.7 ug.mL-1 T07303 C1ZG2U 449087 IC50 > 10000 nM T07303 CCN9D5 3142817 IC50 = 1000 nM T07303 CFW19M 5329009 IC50 = 2400 nM T07303 CDQ3M7 5359485 IC50 = 1.3 ug.mL-1 T07303 C54BYP 5360741 IC50 = 0.96 ug.mL-1 T07303 CUPQ08 6539985 IC50 = 13 nM T07303 CMEZ23 6540005 IC50 = 87 nM T07303 CG17TN 6914611 IC50 > 50000 nM T07303 C7E2QK 6914613 IC50 > 50000 nM T07303 C9TAL6 9826308 IC50 = 92 nM T07303 C7TA9J 10113568 IC50 = 7.586 nM T07303 CIV15Q 10113978 IC50 = 46 nM T07303 C7SFI1 10296883 IC50 = 4600 nM T07303 C8RD3V 10301884 IC50 > 10000 nM T07303 C7HBP6 10429593 IC50 > 10000 nM T07303 CBOP58 11293798 Ki > 10000 nM T07303 C26BZX 11362471 Ki > 10000 nM T07303 CWXB93 11397177 Ki > 10000 nM T07303 CG3BZ9 11517980 IC50 = 8 nM T07303 CL7X4Q 11530963 IC50 = 5 nM T07303 CTG83F 11539329 Ki > 7100 nM T07303 CACS26 11561968 Ki > 2000 nM T07303 CB91RQ 11589811 IC50 = 667 nM T07303 CA2KX0 11590078 IC50 = 4 nM T07303 CM65QP 11590120 IC50 = 29 nM T07303 CMIL86 11590363 Ki > 7100 nM T07303 C7W3TE 11633427 IC50 = 172 nM T07303 C9T6SC 11640926 Ki > 7100 nM T07303 CU0E8O 11690457 Ki > 2000 nM T07303 CUB2N6 11719537 IC50 = 22 nM T07303 CP7AH3 11755812 IC50 = 71 nM T07303 C9JT4S 11847343 IC50 = 19 nM T07303 CHR92S 11858109 IC50 = 5 nM T07303 CQF23E 11952856 IC50 = 11 nM T07303 CC09DE 11955790 IC50 = 123 nM T07303 CM50UH 12000646 EC50 = 60 nM T07303 CDGF78 15282555 IC50 = 2800 nM T07303 CFPW41 16007116 Ki > 7000 nM T07303 CZKD04 16043241 IC50 = 4 nM T07303 C9X4TQ 16043242 IC50 = 68 nM T07303 CP3HS4 16220354 IC50 = 3 nM T07303 CL81VC 21100709 IC50 = 5190 nM T07303 CHU49V 24757938 IC50 = 2 nM T07303 CCPS81 24764502 IC50 > 35000 nM T07303 CQN3Z7 24825710 IC50 = 360 nM T07303 C43HWQ 24883287 IC50 = 2700 nM T07303 C8DA5Q 24883334 IC50 = 4500 nM T07303 C4V9GH 24894117 IC50 = 37 nM T07303 CM6K3X 24894768 IC50 = 3400 nM T07303 CJH19T 24894883 IC50 = 11000 nM T07303 CJ14YB 24894884 IC50 = 8700 nM T07303 CHVU39 24894885 IC50 = 18000 nM T07303 CZ6KD4 24894886 IC50 = 5600 nM T07303 CKBY19 24894887 IC50 = 3200 nM T07303 C57BHF 24894888 IC50 = 3600 nM T07303 CB5TP8 24894992 IC50 = 4800 nM T07303 C32SUJ 24894993 IC50 = 1700 nM T07303 C38TGD 24894994 IC50 = 3200 nM T07303 CP7QT2 24894995 IC50 = 9400 nM T07303 C41SIT 24894996 IC50 = 5300 nM T07303 CFW40U 24894997 IC50 = 2500 nM T07303 CF4N9X 24895100 IC50 = 2500 nM T07303 CN13JF 24899915 IC50 = 1.7 ug.mL-1 T07303 CBWR97 24899916 IC50 = 0.39 ug.mL-1 T07303 C9F2JD 24899917 IC50 > 10 ug.mL-1 T07303 C64MTI 24900160 IC50 = 6.8 ug.mL-1 T07303 CO2I6Q 24900161 IC50 = 3.7 ug.mL-1 T07303 C4EG8R 24993189 IC50 = 587 nM T07303 C3DI7Y 24995523 IC50 = 14 nM T07303 C2ICS7 25065806 IC50 = 151 nM T07303 CX0O5A 25178331 IC50 = 9600 nM T07303 CIG4H0 25178539 IC50 = 4700 nM T07303 CNG96H 25210579 IC50 > 10000 nM T07303 C81UIT 42604010 IC50 = 45000 nM T07303 CJ5U1X 42639664 IC50 = 4 ug.mL-1 T07303 CN8WB9 44189332 IC50 = 417 nM T07303 CYV2D7 44368815 IC50 = 52 nM T07303 C7KZV2 44414322 IC50 = 169 nM T07303 CJM06T 44414347 IC50 = 1573 nM T07303 CBY7D9 44414679 IC50 < 3 nM T07303 C0JF1Z 44414779 IC50 = 23 nM T07303 C4YMI9 44447890 IC50 = 10 nM T07303 C0LY6E 44552561 EC50 = 780 nM T07303 C7KRU3 44552562 IC50 = 140 nM T07303 CC7E4K 44564705 IC50 = 6000 nM T07303 C42ZEW 44564706 IC50 > 10000 nM T07303 C53MCK 44564747 IC50 = 6500 nM T07303 CDI31F 44564748 IC50 = 6900 nM T07303 CA17NT 44564749 IC50 > 10000 nM T07303 CSO9F8 44564751 IC50 = 5200 nM T07303 CM50GS 44564788 IC50 > 10000 nM T07303 C3Q0DX 44564789 IC50 = 2100 nM T07303 CP40XB 44564790 IC50 > 10000 nM T07303 C35NTB 44564791 IC50 > 10000 nM T07303 CJY83G 44564817 IC50 = 7700 nM T07303 CF2D1K 44564819 IC50 = 3400 nM T07303 C3CQ9K 44564820 IC50 > 10000 nM T07303 CI8V2L 44564821 IC50 > 10000 nM T07303 C9PO7J 44564860 IC50 > 10000 nM T07303 C16FJW 44564861 IC50 > 10000 nM T07303 CJ1X9V 44565013 IC50 = 2500 nM T07303 CN2Q3D 44565014 IC50 = 1600 nM T07303 CM2GN3 44565015 IC50 > 10000 nM T07303 CU3RF1 45139989 IC50 > 10000 nM T07303 CQGZ06 45139991 IC50 > 10000 nM T07303 CNI92D 46182735 IC50 = 22.4 nM T07303 CY3HW5 46224684 IC50 = 5800 nM T07303 C8YPN0 46225596 IC50 = 4500 nM T07303 C34JTS 46225597 IC50 = 1700 nM T07303 CGD73B 46225598 IC50 > 10000 nM T07303 CRDY89 46225610 EC50 = 14000 nM T07303 C0JMT8 46225611 IC50 = 1900 nM T07303 CF0D5J 46225612 IC50 = 69 nM T07303 CLZ1O6 46225634 EC50 = 13000 nM T07303 CT70DX 46225640 IC50 = 1500 nM T07303 C6AJ5N 46225647 IC50 = 865 nM T07303 C38BFC 46225657 IC50 = 7100 nM T07303 C1B3KS 46225663 EC50 = 26000 nM T07303 CU46XI 46225664 IC50 = 9300 nM T07303 CO3HS2 46225665 IC50 = 1300 nM T07303 C2UV1S 46225666 EC50 > 10000 nM T07303 CX5B1G 46225667 IC50 = 3000 nM T07303 C2Q9OH 46225668 IC50 > 10000 nM T07303 C8S4QA 46225688 IC50 = 340 nM T07303 CYZV41 46231219 IC50 = 66 nM T07303 C7J5UP 46231220 IC50 = 29.51 nM T07303 CC96GZ 46231221 IC50 = 21 nM T07303 C7ON5A 46233287 IC50 > 10000 nM T07303 CW0P5B 46845702 IC50 = 3010 nM T07303 C7KM0E 46845704 IC50 = 960 nM T07303 C5WC9K 46871765 IC50 = 940 nM T07303 CLS29B 46872626 IC50 > 10000 nM T07303 C2O8RZ 46886323 IC50 = 65 nM T07303 CL5R0D 46888599 IC50 = 2680 nM T07303 C3IE0X 46888601 IC50 = 2170 nM T07303 C1A0XQ 46888603 IC50 = 2050 nM T07303 CB5YQ1 46888635 IC50 = 2530 nM T07303 C6YC4O 46888663 IC50 = 4070 nM T07303 C0AUT8 46888665 IC50 = 2640 nM T07303 CAZT96 46888666 IC50 > 50000 nM T07303 CS4U3P 46888668 IC50 = 1310 nM T07303 CASV10 46888710 IC50 = 1810 nM T07303 CY2TV5 46888712 IC50 = 2270 nM T07303 CX5AL6 46888740 IC50 = 2850 nM T07303 CSWE93 46888742 IC50 = 34570 nM T07303 CW7AR1 46889887 IC50 = 5 nM T07303 CMNK35 46889911 IC50 = 9 nM T07303 CTZ71Y 46898039 IC50 = 0.8 nM T07303 CH5NU2 49798965 IC50 > 1000 nM T07303 C02SVR 49798997 IC50 = 39 nM T07303 C8DA5K 49798998 IC50 = 42 nM T07303 CO18QM 49798999 IC50 = 34 nM T07303 CC8FS1 49799031 IC50 = 12.8 nM T07303 CLNI64 49799032 IC50 = 11 nM T07303 CG7K2D 49799066 IC50 = 92 nM T07303 C27SKR 49799067 IC50 = 146.8 nM T07303 CCX04I 49799068 IC50 = 8.7 nM T07303 CQZC18 49799069 IC50 = 68 nM T07303 C2HA1O 49799301 IC50 = 13 nM T07303 C62OBF 49799302 IC50 > 1000 nM T07303 C1QC4V 49799333 IC50 > 1000 nM T07303 CG3LY7 49799334 IC50 > 1000 nM T07303 CZBW04 49799372 IC50 = 88 nM T07303 CN1M2D 49799373 IC50 = 13 nM T07303 CHIQ50 49799374 IC50 = 5.8 nM T07303 C45FZO 49799375 IC50 = 32.9 nM T07303 CY90BD 49818230 IC50 = 4200 nM T07303 CB0S2P 49842666 IC50 = 1400 nM T07303 C5R6QY 49842669 IC50 > 100000 nM T07303 C0NA9U 49842670 IC50 = 5500 nM T07303 CC7MR2 49842671 IC50 = 17000 nM T07303 CAI20B 49842778 IC50 = 720 nM T07303 CRA74I 49842779 IC50 = 1200 nM T07303 C5RQ7C 50908680 Ki = 680 nM T07303 CD2K4R 50908681 Ki > 1000000 nM T07303 C2Y6QS 50938552 IC50 > 10000 nM T07303 C9NYP4 51036677 IC50 > 10000 nM T07303 C4WRY3 51037112 IC50 > 10000 nM T07303 CRI28Z 51037948 IC50 > 10000 nM T07303 CG9E4A 52942446 Ki > 1000000 nM T07303 C8SJ2Q 52942862 Ki > 1000000 nM T07303 CLO46D 52944812 Ki = 9390 nM T07303 CI6GX2 52948511 Ki = 1090 nM T07303 CWA74O 52949707 Ki = 1090 nM T07303 C2P3OT 53316977 IC50 = 5800 nM T07303 CX59LD 53320915 IC50 = 65000 nM T07303 CZY0J7 53323592 IC50 = 1600 nM T07303 CCKD48 53324892 IC50 > 100000 nM T07303 C8NA4L 53384644 IC50 > 30000 nM T07303 CE1ZK6 54759168 IC50 > 10000 nM T07303 C8AB1J 54759606 Ki < 0.3 nM T07303 CR50TJ 56835147 IC50 = 9.6 nM T07303 CP58NG 56954518 IC50 = 9 nM T07303 C4WE9B 57391179 IC50 = 51 nM T07303 CY10TP 57391180 IC50 = 101 nM T07303 CU3DM9 57391295 IC50 > 10000 nM T07303 CU7J9C 57393063 IC50 < 5 nM T07303 CD4HS3 57393074 IC50 = 177 nM T07303 CS60KL 57393075 IC50 > 10000 nM T07303 CWMT98 57394785 IC50 > 10000 nM T07303 C9PY4Q 57394798 IC50 = 175 nM T07303 C3F9VS 57394799 IC50 = 3063 nM T07303 C4CN6V 57396453 IC50 = 25 nM T07303 CCT58R 57396454 IC50 = 453 nM T07303 CXA5Z9 57396541 IC50 = 57 nM T07303 CPAH35 57396542 IC50 = 35 nM T07303 CY8U1Q 57396557 IC50 = 8 nM T07303 CWV96N 57398329 IC50 = 39 nM T07303 C8K1WJ 57398330 IC50 = 0.2 nM T07303 CBK02S 57399984 IC50 = 7 nM T07303 CNU4I7 57399985 IC50 = 30 nM T07303 CD9KF3 57399986 IC50 = 282 nM T07303 C0BA7P 57401686 IC50 = 485 nM T07303 CH56JP 57401785 IC50 = 31 nM T07303 C7YMG1 57401804 IC50 = 6144 nM T07303 C20ZAX 57401805 IC50 = 209 nM T07303 C15YQW 57401806 IC50 = 128 nM T07303 CY5TJ9 57401807 IC50 < 5 nM T07303 C4L0SA 57401808 IC50 = 12 nM T07303 C4J0OD 57403506 IC50 = 0.4 nM T07303 CN0M3Z 57403518 IC50 = 1009 nM T07303 CZSM95 57412684 IC50 = 3700 nM T07303 C8R4FE 57991377 IC50 = 554.5 nM T07303 CI50KU 58167984 IC50 = 867 nM T07303 C1MR8Q 60097495 IC50 > 1000 nM T07303 C7MLW5 60182318 IC50 = 0.1 nM T07303 CV63UL 67240318 IC50 > 10000 nM T07303 CCN01X 71547862 IC50 > 10000 nM T07303 CB64IQ 72194525 IC50 = 4.5 nM T07303 CGDB30 74538658 IC50 = 30 nM T07303 C29EZO 76871930 IC50 = 600 nM T07303 CPG3A5 86302574 IC50 > 30000 nM T07303 CY0UC4 90645194 IC50 > 10000 nM T07303 CP34KC 90664681 IC50 = 1660 nM T07303 CK3IS4 90664930 IC50 = 2220 nM T07303 CY7BI2 118706214 IC50 > 10000 nM T07303 C3KLI5 118723185 IC50 = 5000 nM T07303 C8U0ZH 118737468 IC50 = 4.55 nM T07303 C4X7SD 122192466 IC50 = 1188 nM T07303 CNX0Q2 122193763 IC50 = 47 nM T07303 CWV0C3 122193764 IC50 = 1980 nM T07303 CSG98Y 122193765 IC50 = 420 nM T07303 CCLQ75 122193769 IC50 = 7 nM T07303 CXDR48 122193770 IC50 = 6 nM T07303 CPA8C5 122193773 IC50 = 1020 nM T07303 C2LAM7 126591927 IC50 = 72 nM T07303 C8TB3R 127041351 IC50 = 4 nM T07303 C40WEH 127041352 IC50 = 5.5 nM T07303 CUO0C5 132156633 IC50 > 10000 nM T07303 C6OMB1 132204257 IC50 = 141 nM T07303 CJ04HZ 132585195 IC50 = 72 nM T07303 CI2YE9 132606873 IC50 = 114.5 nM T07303 CLCO61 135398510 IC50 = 3 nM T07303 CK9D4A 135428921 IC50 = 520 nM T07303 CS63IO 135476717 IC50 = 13 nM T07303 CRFQ36 135800265 IC50 < 10000 nM T07303 CHA4N2 136013680 IC50 > 10 nM T07303 C1YUD0 136219394 IC50 > 10 nM T07303 CIU8W3 136254389 IC50 > 10 nM T07303 CCM42D 137249694 IC50 = 9.6 nM T07303 CXC69T 137321158 IC50 = 20 nM T07303 C6L3HN 137634634 IC50 = 43 nM T07303 CQMB10 137658515 IC50 = 376 nM T07303 CIWG23 138393067 IC50 = 46 nM T07303 CI1D9F 139600335 IC50 = 8 nM T07303 C34CKN 141523354 IC50 = 183.1 nM T07303 CB3Z1W 145949428 IC50 = 45 nM T07303 C1IX5N 145956333 IC50 = 18.2 nM T07303 C5VSC7 145956704 IC50 = 37 nM T07303 CY54UC 145957309 IC50 = 23.01 nM T07303 CTUF34 145966712 IC50 = 113 nM T07303 C74TYP 145975351 IC50 = 23.6 nM T07303 C7X3WN 155513030 IC50 > 10000 nM T07303 C86HPW 155518524 IC50 > 100000 nM T07303 C3ST0D 155522792 IC50 = 9.2 nM T07303 CXFH76 155523422 IC50 = 1.1 nM T07303 C3UT5M 155535028 IC50 > 10000 nM T07303 C8H1CZ 155536201 IC50 > 10000 nM T07303 CFEZ25 155539618 IC50 = 27 nM T07303 C0HC7V 155540067 IC50 = 190 nM T07303 CA5I7X 155541030 IC50 > 10000 nM T07303 CL7N0Q 155542435 IC50 > 10000 nM T07303 C7NRO6 155545934 IC50 = 9.9 nM T07303 C3VX6K 155547248 IC50 = 23 nM T07303 CW34RN 155549665 IC50 = 14.2 nM T07303 CYO3B0 155554258 IC50 = 17.3 nM T07303 C40IYS 155562258 IC50 = 591 nM T07303 CD2XG9 155564539 IC50 = 5300 nM T07303 CX8I9K 155567999 IC50 = 7.8 nM T07303 D00ERW 44444843 Ki = 6846 nM T07303 D00HVA 11624601 Ki > 7100 nM T07303 D02BXJ 46864270 IC50 = 2.6 nM T07303 D03DZO 11715767 IC50 > 10000 nM T07303 D05NKG 16760286 IC50 = 1000 nM T07303 D06QWO 14824655 IC50 > 10 ug.mL-1 T07303 D07IHM 9823787 IC50 = 2459 nM T07303 D07OXC 11650194 IC50 = 120 nM T07303 D08GBT 71295845 IC50 = 1.2 nM T07303 D08HFG 24809764 IC50 > 10000 nM T07303 D09HVH 135566652 IC50 > 10 nM T07303 D09PTP 57325421 IC50 = 48 nM T07303 D09QBA 23378546 IC50 > 10000 nM T07303 D0A1CM 5281855 IC50 = 1540 nM T07303 D0C2GE 67161540 IC50 = 3.2 nM T07303 D0E7VO 59627005 IC50 = 64 nM T07303 D0EE6A 6398883 IC50 = 18 nM T07303 D0G3SZ 6918469 IC50 > 10 ug.mL-1 T07303 D0IR6U 5494425 IC50 = 690 nM T07303 D0M4QA 56935577 IC50 = 1.3 nM T07303 D0Q3NG 11715520 Ki > 7100 nM T07303 D0Q4EQ 16742063 IC50 = 1100 nM T07303 D0S7IE 11658882 Ki > 7100 nM T07303 D0T8NU 16757525 IC50 > 4000 nM T07303 D0US9O 45275255 IC50 = 40 nM T17863 D0EV6T 54682461 Ki = 2000 nM T17863 D04TSV 9875002 IC50 = 202000 nM T17863 D04ZIJ 5478883 IC50 = 59 nM T17863 CJI39W 3013742 IC50 = 5400 nM T17863 C50ESG 3013755 IC50 = 4100 nM T17863 CX0B5L 9853618 IC50 > 100000 nM T17863 C69KGX 10394329 Ki = 13 nM T17863 CFPX35 11167950 IC50 = 830 nM T17863 CU80VL 11290116 IC50 > 50000 nM T17863 CE6CH3 11583947 IC50 > 50000 nM T17863 CED2Y7 11640634 IC50 > 50000 nM T17863 CE12CX 15018069 Ki = 1240 nM T17863 CI41XT 15126555 Ki = 24 nM T17863 CAY1B5 16090342 IC50 > 50000 nM T17863 CP5G7V 16090348 IC50 > 50000 nM T17863 CMXJ30 23625795 IC50 > 10000 nM T17863 CWF5Z3 25143506 IC50 > 30000 nM T17863 CS7XD5 44321765 Ki = 57 nM T17863 C2OFK8 44321766 Ki = 16 nM T17863 CZ45LH 44322035 Ki > 10000 nM T17863 CQ09YG 44322074 Ki = 69 nM T17863 C3N9LQ 44322075 Ki = 516 nM T17863 CK0BQ2 44322083 Ki > 10000 nM T17863 CNT69K 44322084 Ki = 77 nM T17863 CN58AQ 44322086 Ki > 10000 nM T17863 C1G0FY 44322087 Ki = 185 nM T17863 C98YAJ 44340299 Ki = 3000 nM T17863 C81WYC 44340319 Ki > 6000 nM T17863 CF3A4M 44343168 IC50 = 4000 nM T17863 CT0HM5 44368301 IC50 > 1000000 nM T17863 C73LHB 44371838 IC50 = 4.2 nM T17863 C2PJ4N 59271992 IC50 > 30000 nM T17863 C56CFA 68448803 IC50 > 10000 nM T17863 CD41QM 90662843 IC50 = 33000 nM T17863 CNE41K 90662913 IC50 = 790 nM T17863 C4X5QD 90662917 IC50 = 1070 nM T17863 CBPH47 90662918 IC50 = 910 nM T17863 C8O7AD 90662919 IC50 = 15000 nM T17863 CC2RH7 90662920 IC50 = 27000 nM T17863 C39JYN 90662928 IC50 = 700 nM T17863 CE4HX6 90662931 IC50 = 1240 nM T17863 CB6S7Z 90663445 Ki = 0.1 nM T17863 C2T6BX 90663446 Ki = 1200 nM T17863 C5FOR0 90663447 Ki = 1.5 nM T17863 C72FWD 91929322 Ki > 10000 nM T17863 D0KK6A 15126552 Ki = 27 nM T17863 D0P6RT 10078814 Ki = 11 nM T58454 D04LVK 57379345 IC50 = 260 nM T58454 D0H0EQ 24826799 IC50 = 1.3 nM T58454 D00DRL 44137946 IC50 = 39 nM T58454 D02WVT 25031915 IC50 = 82.5 nM T58454 D03LWG 53235510 IC50 = 1 nM T58454 D05PZB 135398495 IC50 = 1 nM T58454 D07EHV 44814409 IC50 > 10000 nM T58454 D07HPJ 11476171 IC50 = 2700 nM T58454 D0D4VV 46944259 IC50 = 2.6 nM T58454 D0D6XT 118029202 IC50 = 1290 nM T58454 D0E3TC 44259 IC50 = 34 nM T58454 D0H9FR 118295624 Ki = 1.3 nM T58454 D0NW0T 67462786 IC50 = 2.5 nM T58454 D0VF6E 1401 IC50 = 5 nM T58454 D0XT0W 66555680 IC50 = 7.6 nM T58454 D0Z4RC 24756910 IC50 = 3430 nM T58454 D03BNU 59604787 IC50 > 10000 nM T58454 D0T3ME 156422 IC50 = 24000 nM T58454 CPT61U 5328112 IC50 = 130 nM T58454 CZ3LK2 5330387 IC50 = 210 nM T58454 CRU94N 5330388 IC50 = 2360 nM T58454 CDB68F 5330389 IC50 = 1400 nM T58454 C7CX0H 5330390 IC50 > 293 nM T58454 C8E0XS 5330391 IC50 = 326 nM T58454 CW1VX9 5330392 IC50 = 153 nM T58454 CF01JS 5330804 IC50 = 180 nM T58454 C16VXB 9863538 IC50 > 10000 nM T58454 CA94BM 9932979 IC50 = 190 nM T58454 CHI4A7 10113795 IC50 = 3400 nM T58454 CLX54H 11317348 IC50 = 170 nM T58454 CACS26 11561968 Ki > 2000 nM T58454 CU0E8O 11690457 Ki > 2000 nM T58454 CHR92S 11858109 IC50 = 140 nM T58454 C9TU1O 16046126 IC50 > 1000 nM T58454 CD4C3O 23022619 IC50 = 780 nM T58454 CSB9P6 23022656 IC50 = 4600 nM T58454 CN4GO9 23022671 IC50 = 54 nM T58454 CYJ3M6 23022691 IC50 = 200 nM T58454 CDV73P 23022708 IC50 = 40 nM T58454 CT50FB 23022716 IC50 = 130 nM T58454 CJL0B7 23022732 IC50 = 63 nM T58454 CWM83Z 23022836 IC50 = 100 nM T58454 CA3I4T 24753787 IC50 > 50000 nM T58454 CHU49V 24757938 IC50 = 55 nM T58454 C7YG1N 24759534 IC50 = 70 nM T58454 C43HWQ 24883287 IC50 = 4100 nM T58454 C8DA5Q 24883334 IC50 = 2000 nM T58454 CO1AU7 44382037 IC50 > 10000 nM T58454 C9IKS4 44382047 IC50 = 71 nM T58454 C4KA0W 44382048 IC50 = 200 nM T58454 C63MYG 44382259 IC50 = 440 nM T58454 CK2Z0O 44382310 IC50 = 8900 nM T58454 C3LNH9 44382361 IC50 > 1000 nM T58454 C73BAN 44382373 IC50 > 10000 nM T58454 C54PVI 44382411 IC50 = 350 nM T58454 CH2P3B 44382531 IC50 = 71 nM T58454 C02KNS 44382615 IC50 = 23 nM T58454 CRYJ87 44382744 IC50 = 260 nM T58454 C56FIY 44382790 IC50 = 70 nM T58454 CE27NC 44382806 IC50 = 200 nM T58454 CIS1F5 44382807 IC50 > 10000 nM T58454 CW3BP8 44398371 IC50 = 270 nM T58454 CYT37A 46232443 IC50 = 24000 nM T58454 C48ZVW 46232555 IC50 = 6900 nM T58454 CS9B1U 46232556 IC50 = 12000 nM T58454 C0WYM1 46898022 IC50 = 10000 nM T58454 C5ME3S 49806721 IC50 > 50000 nM T58454 C90ANW 50939489 IC50 = 10 nM T58454 CVZU97 51346202 IC50 = 1230 nM T58454 C09SDH 53257410 IC50 > 10000 nM T58454 C4F6SR 53348188 IC50 = 2.29 nM T58454 CM7P3W 53357328 IC50 = 360 nM T58454 C8NA4L 53384644 IC50 > 30000 nM T58454 CPHX64 57325478 IC50 > 50000 nM T58454 CQ9BW4 57325479 IC50 > 50000 nM T58454 CVK0G4 58056356 IC50 > 50000 nM T58454 CXJ63M 59603829 IC50 = 170 nM T58454 CQEU96 59603842 IC50 = 11 nM T58454 CPU2E3 59737752 IC50 = 4433 nM T58454 C1MR8Q 60097495 IC50 > 1000 nM T58454 C9O4GF 66555232 IC50 = 65 nM T58454 CL3EN2 66556938 IC50 = 19 nM T58454 CV63UL 67240318 IC50 > 10000 nM T58454 CO6W9D 68004741 IC50 = 3.6 nM T58454 CB6U7F 68005465 IC50 = 5.2 nM T58454 CK83VI 68005486 IC50 = 41 nM T58454 C1RJ7Y 68005600 IC50 = 21 nM T58454 COX3U9 68005621 IC50 = 9.4 nM T58454 CEXN58 68005732 IC50 = 150 nM T58454 C8I7GC 68293638 IC50 > 10000 nM T58454 C0HA8V 68783839 IC50 = 2 nM T58454 C5DGR9 69036886 IC50 = 591 nM T58454 C9DIK2 71512060 IC50 > 10000 nM T58454 CRX81Q 71575642 IC50 = 1805 nM T58454 C9OQ2I 72710839 IC50 = 493 nM T58454 C2PAK9 73438493 IC50 = 272 nM T58454 CQ5E3H 73707531 IC50 < 1 nM T58454 CBAT06 76071144 IC50 = 930 nM T58454 CRQO23 86293280 IC50 = 369 nM T58454 C4OC7T 86293469 IC50 = 34 nM T58454 CPG3A5 86302574 IC50 > 30000 nM T58454 C1HW4B 89735655 IC50 = 17000 nM T58454 CR1N0E 90367910 IC50 = 0.5 nM T58454 CF27DP 91825767 IC50 = 4 nM T58454 CVB8Q7 118728412 IC50 = 63 nM T58454 CH1B5J 118893306 IC50 = 0.7 nM T58454 C4X7SD 122192466 IC50 > 10000 nM T58454 C1E4AR 122604567 IC50 > 10000 nM T58454 CY30FL 123752658 IC50 = 0.3 nM T58454 CR49HZ 127045733 IC50 < 10 nM T58454 CZG45F 127045746 IC50 = 100.9 nM T58454 C9PNA4 127045747 IC50 = 4.8 nM T58454 CHGQ64 127045748 IC50 = 3.9 nM T58454 C1SG4D 127045749 IC50 = 4.3 nM T58454 C1T6JN 127045945 IC50 = 0.8 nM T58454 CF2U9X 127045946 IC50 = 0.3 nM T58454 C6C0VD 127045973 IC50 = 0.7 nM T58454 C7JN6U 127045974 IC50 < 0.1 nM T58454 C8M5NR 127046432 IC50 = 0.4 nM T58454 C2FO5U 127046442 IC50 < 0.1 nM T58454 CUA4D5 127046443 IC50 = 0.7 nM T58454 CDH30L 127046448 IC50 = 0.6 nM T58454 C7V9LZ 127046449 IC50 = 1.2 nM T58454 CO2ID1 127046609 IC50 = 0.3 nM T58454 C4UBV5 127046610 IC50 = 9 nM T58454 CI5HW2 127046778 IC50 = 3.2 nM T58454 CL9VO8 127047232 IC50 = 0.4 nM T58454 CN2ZV4 127047233 IC50 = 1.3 nM T58454 C56LZX 127047295 IC50 = 0.6 nM T58454 CL5IA8 127047296 IC50 = 0.5 nM T58454 CA95LC 127047297 IC50 = 0.7 nM T58454 CX43YM 127047298 IC50 = 16.9 nM T58454 CS58UX 127047353 IC50 = 2.7 nM T58454 CGV28E 127047354 IC50 = 0.9 nM T58454 CL54JP 127047842 IC50 < 0.1 nM T58454 C6AOY4 127047843 IC50 = 0.7 nM T58454 C6SWY8 127047845 IC50 = 0.9 nM T58454 C9SI5T 127047969 IC50 < 0.4 nM T58454 CUO0C5 132156633 IC50 > 10000 nM T58454 CML72V 132185297 IC50 = 1.1 nM T58454 CM8TC3 132185299 IC50 = 8 nM T58454 CWY58Z 132185302 IC50 = 7.2 nM T58454 CK9W4F 134135741 IC50 = 940 nM T58454 CMA60G 134144799 IC50 = 870 nM T58454 C3MN6B 134144868 IC50 = 920 nM T58454 CEZH84 134146580 IC50 = 450 nM T58454 C1DF4R 134147544 IC50 = 230 nM T58454 C95NCV 134151662 IC50 = 30 nM T58454 CX7YE1 134155961 IC50 = 32 nM T58454 CE38MW 134156584 IC50 = 4.2 nM T58454 CVI25K 134157526 IC50 = 140 nM T58454 CO1IL0 134457555 IC50 > 10000 nM T58454 CB15KN 134457556 IC50 > 10000 nM T58454 CCFS35 134457606 IC50 > 10000 nM T58454 CEAH09 134457612 IC50 > 10000 nM T58454 C1P9KY 134457618 IC50 > 10000 nM T58454 CGAV72 134457621 IC50 = 396.8 nM T58454 CWZ1L4 135316948 IC50 = 2.73 nM T58454 C5B6XD 135316952 IC50 = 2.39 nM T58454 CWEP52 135316962 IC50 = 1.65 nM T58454 CW5KL0 135316982 IC50 = 2.61 nM T58454 C6E5FP 135317017 IC50 = 1.21 nM T58454 CCTW97 135317286 IC50 = 0.84 nM T58454 CH2JK6 135317468 IC50 = 1.58 nM T58454 CFE0X7 135317546 IC50 = 1.62 nM T58454 C0JM1W 135317567 IC50 = 1.77 nM T58454 CI2L5A 135317791 IC50 = 1.45 nM T58454 CJZ59L 135317844 IC50 = 1.39 nM T58454 C45XNW 135318783 IC50 = 3.63 nM T58454 CS63IO 135476717 IC50 = 37 nM T58454 C4WX3I 135486449 IC50 = 13460 nM T58454 CYXU86 136180312 IC50 = 9130 nM T58454 C9MHA4 136180313 IC50 = 9130 nM T58454 CDT7E4 136211077 IC50 = 2 nM T58454 C7PNC4 136243300 IC50 = 15730 nM T58454 CUN1I4 136243344 IC50 = 17710 nM T58454 C68IKN 136243473 IC50 = 8390 nM T58454 CDY18N 136301774 IC50 = 3000 nM T58454 CH4T8M 136961363 IC50 = 9580 nM T58454 C7N8EG 136961364 IC50 = 16110 nM T58454 CRPQ98 136961365 IC50 = 13470 nM T58454 CSZ16N 136961366 IC50 = 6280 nM T58454 CB9D7F 136961367 IC50 = 7620 nM T58454 CEPT42 136961368 IC50 = 6140 nM T58454 C25ERN 137631967 IC50 = 2 nM T58454 CLQT06 137632162 IC50 > 1000 nM T58454 C0J6IC 137633737 IC50 = 1000 nM T58454 CNX0F9 137634126 IC50 = 27 nM T58454 CB35YZ 137634742 IC50 = 56.4 nM T58454 CF7P1V 137635991 IC50 > 1000 nM T58454 C2K8LT 137636345 IC50 > 10000 nM T58454 CUR48O 137636669 IC50 = 250.2 nM T58454 CF7O2C 137636828 IC50 > 10000 nM T58454 CPR60M 137637024 IC50 > 10000 nM T58454 C06JRX 137637094 IC50 = 155.7 nM T58454 CH2OR6 137637188 IC50 > 1000 nM T58454 CMCI72 137638094 IC50 > 10000 nM T58454 C8AI5O 137638529 IC50 = 44.6 nM T58454 CP3SA8 137639345 IC50 > 1000 nM T58454 C7J8FB 137639540 IC50 > 10000 nM T58454 CXM2I8 137640932 IC50 = 2.8 nM T58454 CRQG32 137641135 IC50 = 3 nM T58454 C9FH7X 137641558 IC50 = 108.5 nM T58454 C9WBQ0 137641746 IC50 = 26.3 nM T58454 C5E6NQ 137643062 IC50 > 10000 nM T58454 CY8L5M 137644036 IC50 = 493 nM T58454 CJ2M1O 137644088 IC50 = 2 nM T58454 C0CTB5 137644554 IC50 > 10000 nM T58454 CS3TU7 137644762 IC50 > 10000 nM T58454 C0P1CJ 137644932 IC50 = 35.1 nM T58454 C9B7XU 137645188 IC50 = 50.5 nM T58454 CEO3V1 137645361 IC50 = 100 nM T58454 C09CLU 137646239 IC50 = 100 nM T58454 C79SUZ 137646264 IC50 = 311.9 nM T58454 C7P5AX 137646321 IC50 > 10000 nM T58454 C0YP8D 137646334 IC50 = 16.1 nM T58454 CBK62Y 137646491 IC50 = 6.6 nM T58454 C7CA9N 137646692 IC50 > 10000 nM T58454 C5IB6V 137647631 IC50 = 7 nM T58454 CS3H8E 137647913 IC50 > 1000 nM T58454 CGF7X2 137647982 IC50 = 414 nM T58454 C7EZP8 137649394 IC50 > 10000 nM T58454 CP2N8Y 137649616 IC50 = 16.6 nM T58454 CBK9F7 137650459 IC50 = 35.1 nM T58454 CO4HY7 137650511 IC50 = 280.1 nM T58454 CHSB74 137650627 IC50 > 10000 nM T58454 CRUE07 137651077 IC50 = 9.5 nM T58454 C1DK0P 137651391 IC50 = 4.7 nM T58454 C47VJA 137651444 IC50 = 153.5 nM T58454 CIR94V 137651828 IC50 > 1000 nM T58454 C6EN8I 137652073 IC50 = 293.5 nM T58454 CU5J4G 137652158 IC50 = 56.9 nM T58454 C0MZ1W 137652333 IC50 > 10000 nM T58454 CD7UV3 137652920 IC50 = 71.9 nM T58454 CBAF08 137653174 IC50 > 10000 nM T58454 CTV31U 137653424 IC50 > 1000 nM T58454 C6S2ZA 137654098 IC50 < 4.1 nM T58454 C4B7FC 137655376 IC50 > 1000 nM T58454 CQ85OV 137655810 IC50 > 1000 nM T58454 C01JVI 137656138 IC50 = 72.9 nM T58454 CFWN28 137657383 IC50 = 132.7 nM T58454 CWA62P 137657677 IC50 = 2 nM T58454 CV5H3Z 137657932 IC50 = 8.6 nM T58454 CSC2G0 137658026 IC50 = 2.9 nM T58454 C7SEK1 137658232 IC50 > 10000 nM T58454 CQF74K 137658987 IC50 > 10000 nM T58454 C8DZ6L 137659285 IC50 > 10000 nM T58454 C4DT3V 137659387 IC50 > 1000 nM T58454 CY8B6K 137659396 IC50 > 1000 nM T58454 CD3K9G 137659884 IC50 = 100 nM T58454 C9UMG4 137660300 IC50 = 1000 nM T58454 CS04UY 137660727 IC50 > 1000 nM T58454 CIV31M 137661021 IC50 > 1000 nM T58454 CW9U3A 137661140 IC50 > 10000 nM T58454 C82WHL 137661196 IC50 = 36.2 nM T58454 CK2GY9 137661845 IC50 = 91 nM T58454 CM3UF7 137700779 IC50 > 10000 nM T58454 CSRI06 138547901 IC50 = 1.5 nM T58454 CUXO19 138617501 IC50 = 0.8 nM T58454 CZ2XH5 139187793 IC50 > 10000 nM T58454 CUH2G6 139554482 IC50 = 2.2 nM T58454 CO9P7G 145351804 IC50 = 4.5 nM T58454 C29XUO 145945978 IC50 = 6.6 nM T58454 C15SAP 145949598 IC50 = 6400 nM T58454 CL14YA 145950580 IC50 = 52000 nM T58454 C1AL5N 145952450 IC50 = 800 nM T58454 C2QOE5 145956264 IC50 = 7300 nM T58454 C7MBT6 145957742 IC50 = 5400 nM T58454 CSZ14F 145958261 IC50 = 12000 nM T58454 C93AOR 145980752 IC50 = 363 nM T58454 C03PYD 145986466 IC50 < 1000 nM T58454 CS7TD1 145993995 IC50 > 10000 nM T58454 CN7EF3 145996526 IC50 > 1000 nM T58454 C2MD1Q 155513187 IC50 > 10000 nM T58454 C86HPW 155518524 IC50 = 23000 nM T58454 CL3DV0 155519320 IC50 = 2 nM T58454 CFRQ41 155530069 IC50 = 1.9 nM T58454 CS69CA 155532132 IC50 = 39.2 nM T58454 CX37HC 155537699 IC50 > 1000 nM T58454 D02BXJ 46864270 IC50 = 1.5 nM T58454 D04NGS 5330790 IC50 = 220 nM T58454 D06FFZ 91827382 IC50 = 4 nM T58454 D06HVH 54613583 IC50 > 10000 nM T58454 D07OXC 11650194 IC50 > 1000 nM T58454 D09TNR 9850161 IC50 = 69 nM T58454 D0H1OK 11562302 Ki = 493 nM T58454 D0IR6U 5494425 IC50 = 940 nM T58454 D0U3NI 53246941 IC50 = 320 nM T33584 D00ENY 33032 Ki = 1360 nM T33584 D03CNS 2910 EC50 = 1000 nM T33584 D0U3ED 9924495 IC50 = 243 nM T33584 D02VKC 3272524 Ki = 1600 nM T33584 D0B0NQ 127894 Ki = 9200 nM T33584 D0M7MW 126758 EC50 = 28000 nM T33584 COC91V 10255 Ki = 7449 nM T33584 C6T4AH 167842 Ki = 92 nM T33584 CC0E1V 447081 Ki = 5.22 nM T33584 CNBI79 447083 EC50 = 270 nM T33584 CO28NU 447407 EC50 = 22000 nM T33584 C5LW8Q 973101 IC50 = 2970 nM T33584 C1EP3D 2733518 Ki = 170 nM T33584 CWK7X4 4694356 Ki = 130 nM T33584 C3JXD9 5289518 EC50 = 5200 nM T33584 C5Z8VG 6324635 Ki > 10000 nM T33584 CBUK20 6451148 EC50 = 21000 nM T33584 CVW4L3 9795654 Ki = 29 nM T33584 C9TLQ4 9861035 Ki > 10000 nM T33584 C3WNM6 9902629 EC50 = 2880 nM T33584 CFV03Y 9926589 Ki = 134000 nM T33584 CFC2P8 9928016 EC50 = 5650 nM T33584 CB91SA 10122460 Ki = 168 nM T33584 C7Q1MJ 10132082 IC50 > 100000 nM T33584 CME06Q 10155236 EC50 = 910 nM T33584 CRJ2T0 10219992 Ki = 1100 nM T33584 CH2O3K 10270530 EC50 = 660 nM T33584 C5PD0H 10330442 Ki = 700 nM T33584 CFKJ76 10352480 Ki = 185 nM T33584 C7GIJ3 10398361 Ki > 100000 nM T33584 C1N2VM 10420002 Ki = 150 nM T33584 CXE7F5 10541731 Ki > 10000 nM T33584 CN20QX 10598970 Ki = 65 nM T33584 C0O6ZI 10658567 EC50 > 3000000 nM T33584 CJZ04V 11096831 Ki = 279 nM T33584 CQ38WM 11219775 Ki = 5150 nM T33584 CGRT02 11288627 Ki = 145 nM T33584 CHUX80 11818375 Ki = 10000 nM T33584 CDGZ79 11820131 Ki = 113400 nM T33584 CGO18D 14608128 Ki = 22000 nM T33584 CQ2YP8 16659202 EC50 = 500000 nM T33584 CDZ2E6 18713992 EC50 = 5650 nM T33584 C1OW7A 24755637 EC50 = 18500 nM T33584 CFLR45 24850230 EC50 = 4100 nM T33584 C4U7OS 44152410 Ki = 65 nM T33584 CW9TR7 44346780 Ki = 7.1 nM T33584 C64ELF 44346789 Ki = 240 nM T33584 CQJW06 44346790 Ki = 163 nM T33584 C15MPO 44346798 Ki = 73.9 nM T33584 CVJA46 44368884 Ki = 78 nM T33584 CH5ZV3 44368885 Ki = 64 nM T33584 CY67GS 44368886 Ki = 88 nM T33584 C0SN1C 44368895 Ki = 68 nM T33584 C0QG8D 44368910 Ki = 100 nM T33584 C64QPC 44369047 Ki = 350 nM T33584 CHAQ75 44369048 Ki = 90 nM T33584 CIOF54 44369061 Ki = 38 nM T33584 CL4I1Y 44369062 Ki = 110 nM T33584 C9F0SZ 44369077 Ki = 220 nM T33584 CM0LI2 44369235 Ki = 110 nM T33584 C4U2TZ 44369248 Ki = 130 nM T33584 CES5P3 44369251 Ki = 250 nM T33584 C2P9GS 44369283 Ki = 3.3 nM T33584 CCIZ47 44369293 Ki = 130 nM T33584 C60TGF 44369295 Ki = 168 nM T33584 C0RAW6 44369306 Ki = 410 nM T33584 C9X3SO 44369308 Ki = 468 nM T33584 C38HPQ 46886654 EC50 = 258 nM T33584 C6HJZ0 52941898 EC50 < 10000 nM T33584 C82PJH 74223604 IC50 = 65.3 nM T33584 C5IXE2 74763075 IC50 = 1790 nM T33584 C1O9RY 118536491 IC50 = 9260 nM T33584 CS12LE 118536551 IC50 = 83300 nM T33584 CT7GO1 127048574 IC50 = 615 nM T33584 CHY6N8 127048930 IC50 = 50.9 nM T33584 CN5DS4 127048931 IC50 = 53.9 nM T33584 CLT8S9 127048932 IC50 = 2820 nM T33584 CNB16I 127049260 IC50 = 22 nM T33584 CPU14C 127049895 IC50 = 70 nM T33584 CN3AM1 127050488 IC50 = 53.6 nM T33584 CUFT19 127052038 IC50 = 147 nM T33584 C8VWC5 127052039 IC50 = 353 nM T33584 CGUB79 127052040 IC50 = 83300 nM T33584 C5Q6ZI 137638800 Ki = 6400 nM T33584 C03KAU 155519563 EC50 > 1000000 nM T33584 CW4H5L 155522120 EC50 > 1000000 nM T33584 D01DMS 447196 Ki = 163 nM T33584 D03RGP 1221 Ki = 22 nM T33584 D04SMQ 440053 Ki = 386 nM T33584 D09LXQ 126569 Ki = 14.7 nM T33584 D0KD6O 5288598 EC50 = 4500 nM T33584 D0N1CL 9799478 IC50 > 100000 nM T33584 D0O7OE 122294 IC50 = 350 nM T33584 D0SB9H 119582 IC50 = 40 nM T33584 D0T5SU 158397 Ki = 21.9 nM T75643 D0C4RB 36314 IC50 = 7943.28 nM T75643 D0O5WP 148124 IC50 = 5011.87 nM T75643 CORM50 584781 IC50 > 20000 nM T75643 C2VZH3 647508 IC50 > 20000 nM T75643 C43VDF 743900 IC50 = 11900 nM T75643 C3VK0C 746711 IC50 > 20000 nM T75643 CF92JY 755364 IC50 > 20000 nM T75643 C27RMY 814607 IC50 = 18100 nM T75643 CYOS57 909915 IC50 = 750 nM T75643 CQ04VL 1088429 IC50 > 20000 nM T75643 C83ECX 1088431 IC50 > 20000 nM T75643 C0BJ4Y 1088435 IC50 = 3800 nM T75643 CBP2S9 1088438 IC50 > 20000 nM T75643 CSY32B 1088439 IC50 = 19900 nM T75643 CP40AO 1106348 IC50 > 20000 nM T75643 CWG9X3 1106353 IC50 = 3540 nM T75643 C31QOG 1106356 IC50 = 1620 nM T75643 CPM4V8 1106360 IC50 = 570 nM T75643 CRN6H2 1106361 IC50 = 400 nM T75643 CKLU94 1142837 IC50 = 1850 nM T75643 C5JTM8 1360138 IC50 = 780 nM T75643 CYO14C 3025920 IC50 > 20000 nM T75643 CJ72HY 3025945 IC50 > 20000 nM T75643 CETX38 5310346 IC50 = 12700 nM T75643 C0ZI8N 14783456 IC50 = 6450 nM T75643 CW6RP7 15992998 IC50 > 20000 nM T75643 C5C2LS 15994862 IC50 > 20000 nM T75643 C1DEF3 15996790 IC50 = 1750 nM T75643 C8Y9WJ 16000292 IC50 > 20000 nM T75643 CNIO43 16002787 IC50 = 1550 nM T75643 C4ZPG6 16021204 IC50 = 3290 nM T75643 C5PUD1 19062910 IC50 > 20000 nM T75643 C1ZAB6 20853147 IC50 = 8270 nM T75643 CR0EV3 20853151 IC50 = 3720 nM T75643 C65QXZ 20853209 IC50 > 20000 nM T75643 CGW08K 20901603 IC50 = 3630 nM T75643 C5VKZ1 20901630 IC50 = 17400 nM T75643 CGJ05B 20901660 IC50 = 7900 nM T75643 CG9Y7Z 20901691 IC50 = 390 nM T75643 C0CGA3 26528163 IC50 > 20000 nM T75643 CYV4Q6 41455001 IC50 > 20000 nM T75643 CX9B7O 41455005 IC50 > 20000 nM T75643 C9EC6T 42370913 IC50 > 20000 nM T75643 CH49XR 44182107 IC50 > 20000 nM T75643 CJ6G9A 44182108 IC50 > 20000 nM T75643 CEY1Z0 44182132 IC50 = 1410 nM T75643 CNS3C2 44182143 IC50 = 600 nM T75643 C2OMP6 44182144 IC50 = 1580 nM T75643 CA9GE5 44182145 IC50 = 200 nM T75643 C65SAT 44182146 IC50 = 3450 nM T75643 C8R2GZ 44182147 IC50 > 20000 nM T75643 CY02GM 44182148 IC50 > 20000 nM T75643 CU1X7V 44182149 IC50 = 260 nM T75643 CQL3Y2 44182150 IC50 > 20000 nM T75643 C6AUS5 44229052 IC50 > 20000 nM T75643 CG6YQ2 44229053 IC50 = 3580 nM T75643 CH6QI1 44229054 IC50 > 20000 nM T75643 CJWQ24 44229055 IC50 = 30 nM T75643 C7QTA4 44229056 IC50 > 20000 nM T75643 CEA0F8 44229057 IC50 > 20000 nM T75643 CVX8C7 44229058 IC50 > 20000 nM T75643 CU98HG 44229059 IC50 > 20000 nM T75643 CZ2X0O 44229060 IC50 > 20000 nM T75643 CT28PV 44229066 IC50 > 20000 nM T75643 C3PXS0 44229067 IC50 > 20000 nM T75643 COAV34 44236880 IC50 > 20000 nM T75643 CDNB26 44251466 IC50 > 20000 nM T75643 CX84MR 44251468 IC50 = 8450 nM T75643 CA9CN4 44251469 IC50 > 20000 nM T75643 C9XJI7 44251470 IC50 = 9240 nM T75643 CAD8P0 44251474 IC50 > 20000 nM T75643 CA5JC4 44251475 IC50 > 20000 nM T75643 CNP1T4 44412097 IC50 = 23400 nM T75643 CC1AV6 44543518 IC50 > 20000 nM T75643 C1ELK2 70683344 IC50 > 20000 nM T75643 CPD08T 70693845 IC50 > 20000 nM T75643 CH29GF 71258526 IC50 = 4 nM T75643 CS79JV 117889777 IC50 > 10000 nM T75643 CCL2R0 117907988 IC50 > 10000 nM T75643 C46GHP 117908214 IC50 > 10000 nM T75643 C7SK6U 117908215 IC50 > 10000 nM T75643 CBF7C8 118711983 IC50 > 10000 nM T75643 C2TE9N 118711985 IC50 > 10000 nM T75643 CWM9U7 127047056 EC50 = 2880 nM T75643 C1LDN8 137631490 IC50 = 590 nM T75643 CE73UJ 137631857 IC50 = 4020 nM T75643 C5DIX0 137632307 IC50 = 1190 nM T75643 CN6UQ7 137632365 EC50 = 247 nM T75643 CX1T9D 137632432 IC50 = 1580 nM T75643 CN43SO 137632600 IC50 = 3550 nM T75643 CE5Y3X 137632757 EC50 = 172 nM T75643 CZ29XV 137633122 IC50 = 4160 nM T75643 C4V3EU 137635387 EC50 = 223 nM T75643 C7WC0M 137635525 IC50 = 1320 nM T75643 C4PC1X 137636354 EC50 = 121 nM T75643 CB7JM9 137636367 IC50 = 3790 nM T75643 C2D8EO 137636592 IC50 = 3780 nM T75643 CS9P3G 137637882 IC50 = 2080 nM T75643 C1ZCB7 137638553 IC50 = 2510 nM T75643 CRY36U 137639197 IC50 = 2880 nM T75643 CE5WD2 137639318 IC50 = 7140 nM T75643 CU31EO 137640364 IC50 = 1500 nM T75643 CP6HO8 137641104 EC50 = 472 nM T75643 CXO01A 137642351 IC50 = 900 nM T75643 CH85VU 137643081 IC50 = 3410 nM T75643 CY4DU3 137643953 EC50 = 276 nM T75643 C1H9WD 137644120 IC50 = 870 nM T75643 CEI6X7 137644484 EC50 = 46 nM T75643 C3NDC2 137645474 IC50 = 940 nM T75643 C36RLH 137645722 EC50 = 2790 nM T75643 C0D9ZT 137645928 IC50 = 2990 nM T75643 CZ92HB 137646848 IC50 = 3100 nM T75643 CI0TP1 137647587 EC50 = 777 nM T75643 C3ZWY0 137650229 IC50 = 810 nM T75643 CH78YX 137652947 IC50 = 2270 nM T75643 COU32W 137653192 IC50 = 1020 nM T75643 CJQT49 137653516 IC50 = 2390 nM T75643 CA9R3V 137653573 EC50 = 172 nM T75643 C9CY3A 137655127 IC50 = 5050 nM T75643 CHC9X4 137655226 IC50 = 2280 nM T75643 C8NA1R 137656826 IC50 = 9510 nM T75643 CY0V9Z 137656864 IC50 = 1700 nM T75643 C3ZS8Y 137657750 IC50 = 1240 nM T75643 CT28EF 137660858 IC50 = 420 nM T75643 CF50JU 137661124 EC50 = 388 nM T75643 CAWU53 137661379 EC50 = 6980 nM T75643 C5WJ0C 155521741 IC50 > 25000 nM T75643 CGN5P7 155529528 IC50 = 16900 nM T75643 CZ0NQ1 155536959 IC50 = 9040 nM T75643 CQT7U2 155546687 IC50 = 24600 nM T75643 CY72AR 155566972 IC50 = 12600 nM T75643 D05UGC 451714 EC50 = 46 nM T99402 D00ENY 33032 Ki = 1400 nM T99402 D0DG8W 135565465 EC50 = 79 nM T99402 D0D4OW 57338826 EC50 > 25000 nM T99402 D0U5CS 213056 EC50 > 100000 nM T99402 C0MLE4 1217 Ki > 1000000 nM T99402 CL8RX5 1222 Ki > 1000000 nM T99402 COM10L 1297 IC50 > 1000000 nM T99402 CSM0F5 5115 IC50 > 1000000 nM T99402 CZBT42 73537 EC50 > 1000000 nM T99402 CBN21A 82516 EC50 > 10000 nM T99402 C9H6OS 92136 EC50 > 3000000 nM T99402 CB15YI 125799 EC50 = 7900 nM T99402 CC75PS 126582 EC50 = 4400 nM T99402 CJ6FG7 140002 EC50 > 10000 nM T99402 C34YGT 173564 EC50 > 1000000 nM T99402 CUT07K 177491 Ki = 53000 nM T99402 CF3QI1 282652 EC50 > 5000 nM T99402 CQC9T2 308065 EC50 > 5000 nM T99402 CU3Y4Q 356458 EC50 > 30000 nM T99402 C37ROZ 439282 Ki > 1000000 nM T99402 CO9KU6 443586 Ki > 1000000 nM T99402 C4HCK5 729510 EC50 = 1400 nM T99402 CMT60X 738280 EC50 > 10000 nM T99402 CWS65Z 780819 EC50 > 5000 nM T99402 CM3EO2 836051 EC50 = 4100 nM T99402 CS03BX 869104 EC50 > 10000 nM T99402 CHT57G 871161 EC50 > 10000 nM T99402 CMO9N5 970725 EC50 > 10000 nM T99402 CJQ14R 1012759 EC50 = 5960 nM T99402 CH9XM0 1092658 EC50 = 1170 nM T99402 C1G4VC 1092661 EC50 = 977 nM T99402 C5L0QE 1314024 EC50 = 1440 nM T99402 C4CO5M 1491741 EC50 > 30000 nM T99402 CNI89V 1617110 Ki = 1000000 nM T99402 CB3UZ6 2306530 EC50 > 5000 nM T99402 C6N9EZ 2318321 EC50 > 10000 nM T99402 CDA96S 2441036 IC50 = 4.898 nM T99402 CQP7L1 2442621 EC50 = 1100 nM T99402 CF8DZ9 2445811 IC50 = 10.4 nM T99402 CH2CF8 2447227 EC50 > 5000 nM T99402 CZV0P5 3246152 Ki = 470000 nM T99402 C3HJK8 3525815 EC50 = 220 nM T99402 CC1SN2 3586321 EC50 = 765 nM T99402 CLB94I 4043841 EC50 = 3200 nM T99402 C2S0AR 4066845 EC50 = 226 nM T99402 C6VN4X 4302961 EC50 = 40000 nM T99402 CX3C1G 4338220 EC50 > 10000 nM T99402 COJV81 4521898 EC50 > 10000 nM T99402 CWG1D7 4644726 EC50 = 1400 nM T99402 C3KBW4 4657221 EC50 > 10000 nM T99402 C05WNA 5310956 Ki = 50000 nM T99402 CZT9U2 5916431 EC50 = 7800 nM T99402 C3RTI9 6348408 EC50 = 5940 nM T99402 C7J6KQ 6604704 EC50 = 48000 nM T99402 CD68LI 6604795 Ki > 1000000 nM T99402 CBIK80 6604819 EC50 = 9000 nM T99402 C6QSA9 7157252 Ki > 280000 nM T99402 CTB90X 8403638 EC50 = 2100 nM T99402 CL8JI1 9837114 EC50 > 1000000 nM T99402 CH54PF 9991661 Ki > 280000 nM T99402 C0GN6F 10012356 Ki > 1000000 nM T99402 CQJP31 10012681 Ki > 1000000 nM T99402 CAU7N4 10059959 Ki > 280000 nM T99402 CH6LU7 10103891 EC50 > 1000000 nM T99402 C8H3UO 10176324 EC50 > 100000 nM T99402 C9XQK6 10198133 EC50 > 100000 nM T99402 CL4NP9 10198359 EC50 = 20000 nM T99402 CAZ8P0 10198574 Ki > 280000 nM T99402 CFDX64 10241509 EC50 > 300000 nM T99402 CUA94S 10262421 EC50 = 17000 nM T99402 CZ7A5Y 10263168 Ki > 1000000 nM T99402 CX12HM 10330132 Ki > 1000000 nM T99402 CZ09YG 10358265 IC50 > 300000 nM T99402 CQ1L0O 10359073 Ki > 300000 nM T99402 C6MTC4 10374869 EC50 > 1000000 nM T99402 C09LUW 10375719 EC50 > 30000 nM T99402 CYL91R 10456810 IC50 = 11410 nM T99402 C3KHU7 10465017 EC50 > 1000000 nM T99402 CK9MN4 10465478 EC50 > 1000000 nM T99402 CO9MK3 10489913 Ki > 280000 nM T99402 C34LSX 10489914 Ki > 280000 nM T99402 CU9BA6 10513894 Ki > 280000 nM T99402 CQGZ24 10513895 Ki > 280000 nM T99402 CYC9W8 10513896 Ki > 280000 nM T99402 CH9VN3 10560963 EC50 > 1000000 nM T99402 C57GCR 10656383 Ki = 8800 nM T99402 C8FP7I 10681240 Ki > 280000 nM T99402 CC6T7Z 10704895 Ki > 280000 nM T99402 CC7JP9 10704896 Ki > 280000 nM T99402 CC2PB0 10752213 Ki > 280000 nM T99402 C27KWL 10752214 Ki > 280000 nM T99402 CQTF38 10775369 EC50 = 1000000 nM T99402 C9BK1A 10846649 EC50 = 23000 nM T99402 CASI54 11768848 EC50 > 1000000 nM T99402 C96YUT 11820180 Ki > 1000000 nM T99402 CZU3D1 13285567 EC50 = 2000 nM T99402 CRW7L0 13302355 EC50 = 6900 nM T99402 CD0XJ3 13401655 EC50 = 800 nM T99402 CU6I3M 13435908 EC50 > 30000 nM T99402 CWVF38 14320996 EC50 > 30000 nM T99402 CMG53S 14590355 EC50 = 5800 nM T99402 CDI9O6 14842361 EC50 = 580 nM T99402 CJCD94 15078062 EC50 = 20000 nM T99402 CSW38G 15420544 EC50 > 10000 nM T99402 CZ8PK5 15840277 EC50 > 1000000 nM T99402 CJS57V 16061421 EC50 = 150 nM T99402 C6Q4GL 16747847 EC50 = 720 nM T99402 CM7JD0 16747848 EC50 = 1850 nM T99402 CWU3X9 16748099 EC50 = 580 nM T99402 C4TZY6 17017653 EC50 = 4600 nM T99402 C04GUC 17758443 Ki > 300000 nM T99402 C0Z2XO 17758444 Ki > 300000 nM T99402 CGZF13 17758445 Ki > 300000 nM T99402 C1GSZ4 17758449 Ki > 300000 nM T99402 CZW76I 17758450 Ki > 300000 nM T99402 CT64UF 17758554 Ki > 300000 nM T99402 C3X6WB 17758555 Ki > 300000 nM T99402 C1AD2J 17758556 Ki > 300000 nM T99402 CH6SW3 18084474 IC50 > 30000 nM T99402 CS5B7A 18138918 IC50 > 30000 nM T99402 CWEO80 18756981 Ki = 88000 nM T99402 CN84GO 22037226 EC50 = 2900 nM T99402 CRGH47 22565221 IC50 = 13.8 nM T99402 C0K9DR 22884216 IC50 > 1000000 nM T99402 C0Y4BP 24209760 EC50 > 10000 nM T99402 CI9FL7 24779948 EC50 = 22000 nM T99402 CJR05E 24780088 EC50 = 8000 nM T99402 CW3S6A 24780089 EC50 > 100000 nM T99402 CQ1S9T 24780091 EC50 = 15000 nM T99402 C5OQ7F 24780092 EC50 = 59000 nM T99402 C7F4YL 24780225 EC50 = 4900 nM T99402 C6XLF5 24905646 EC50 > 100000 nM T99402 CFI54P 24905647 EC50 > 100000 nM T99402 CM53FS 25138329 EC50 = 13 nM T99402 CL34WA 25239622 EC50 > 30000 nM T99402 CC1H5I 26187503 EC50 = 372 nM T99402 CTU79Z 30268259 EC50 > 10000 nM T99402 CSG81W 38032499 EC50 > 5000 nM T99402 CE2RH1 40605829 EC50 = 2700 nM T99402 C67KCO 42413689 EC50 > 10000 nM T99402 CJ06RP 42644786 IC50 = 31.6 nM T99402 CKLZ72 42644790 IC50 = 89.2 nM T99402 CEZM36 42644808 EC50 = 56 nM T99402 CP1BQ9 42645256 EC50 > 10000 nM T99402 CK9LI7 44189736 EC50 > 5000 nM T99402 CX64NZ 44189737 EC50 > 10000 nM T99402 CA1W7G 44189738 EC50 > 10000 nM T99402 CK0X9W 44189740 IC50 = 4.6 nM T99402 CNF72Q 44190035 IC50 > 10000 nM T99402 C9L3OI 44191097 EC50 > 10000 nM T99402 CZE38P 44191098 EC50 > 10000 nM T99402 CY7MU1 44191099 EC50 = 2800 nM T99402 CYB78L 44191178 EC50 = 560 nM T99402 C61DUQ 44191179 EC50 > 10000 nM T99402 CO2L5A 44191180 EC50 = 1500 nM T99402 CQH38F 44282281 EC50 = 86000 nM T99402 C0QF7N 44282403 EC50 = 27000 nM T99402 CL13FV 44302605 IC50 > 300000 nM T99402 C03QML 44302608 IC50 > 300000 nM T99402 C2H6QV 44302609 IC50 > 300000 nM T99402 CP1QS5 44302686 IC50 > 300000 nM T99402 C0V9DN 44302818 IC50 > 300000 nM T99402 CDM1P2 44302819 IC50 > 300000 nM T99402 C1GV9Q 44302837 IC50 > 300000 nM T99402 C1FJU0 44302855 IC50 > 300000 nM T99402 C34AVQ 44302856 IC50 > 300000 nM T99402 CKL1M8 44302930 IC50 > 300000 nM T99402 CFTA38 44322537 Ki > 100000 nM T99402 C7E8SH 44322745 Ki > 1000000 nM T99402 CWV7F0 44322840 Ki = 22000 nM T99402 CGL0Z3 44322843 Ki > 1000000 nM T99402 C2SKJ1 44322921 Ki = 23000 nM T99402 CR1OL6 44328753 IC50 = 10080 nM T99402 CUA80G 44328850 IC50 = 62850 nM T99402 CX0Y4F 44329029 IC50 = 20120 nM T99402 C76LOU 44329031 IC50 = 12530 nM T99402 CCV4N5 44329032 IC50 = 9450 nM T99402 CDP86T 44329033 IC50 = 8680 nM T99402 C9V5XC 44329042 IC50 = 60350 nM T99402 CHV03D 44338561 EC50 > 3000000 nM T99402 CJ9WM4 44551744 EC50 = 4900 nM T99402 C9H1GP 44568312 EC50 > 100000 nM T99402 CZG3T6 44569826 Ki > 1000000 nM T99402 CJ28TF 44569827 Ki > 1000000 nM T99402 CFZ64A 44569859 Ki > 1000000 nM T99402 CUW74T 44569860 Ki > 1000000 nM T99402 C2IKO1 44569861 Ki > 1000000 nM T99402 CADV97 44569862 Ki > 1000000 nM T99402 CUC84P 44572061 EC50 > 10000 nM T99402 C2JIC9 44572112 EC50 > 10000 nM T99402 CTM81C 44572113 EC50 = 1400 nM T99402 CFAM64 45082292 EC50 > 1000000 nM T99402 C5TB0R 45101485 EC50 = 950 nM T99402 CS1V2C 45110131 EC50 = 59.4 nM T99402 C3YL0X 45110133 EC50 = 50.4 nM T99402 CUBR32 45110136 IC50 = 11 nM T99402 C5DW4S 45110506 IC50 = 12 nM T99402 C7NFZ1 45110765 EC50 = 674 nM T99402 C50SAB 45111049 EC50 = 177 nM T99402 CIA3C0 45111050 EC50 = 159 nM T99402 CYW84I 45111051 EC50 = 1030 nM T99402 C74INP 45111509 EC50 = 206 nM T99402 C9L8TB 45484609 EC50 = 10000 nM T99402 CZ72DU 45484614 EC50 = 2000 nM T99402 CRSA05 45484621 EC50 = 9600 nM T99402 C3W6IZ 45484623 EC50 = 3100 nM T99402 CF4I3N 45484637 EC50 = 10000 nM T99402 CL92SD 45484642 EC50 = 2000 nM T99402 C47WVX 45484645 EC50 > 10000 nM T99402 COK92G 46182708 EC50 = 27 nM T99402 C31PAF 46700737 EC50 = 220 nM T99402 CD0RK2 46836497 EC50 = 910 nM T99402 C2Y9PB 46836565 EC50 = 140 nM T99402 C27HJR 46836566 EC50 = 750 nM T99402 C1GJK4 46836635 EC50 = 650 nM T99402 CG4S8W 46836637 EC50 = 1100 nM T99402 CI7R8M 46836709 EC50 = 105 nM T99402 CGS4F2 46836713 EC50 = 7 nM T99402 CD0Q1M 46836714 EC50 = 65 nM T99402 C30UTN 46836715 EC50 = 3000 nM T99402 CD26FP 46836786 EC50 = 51 nM T99402 C8VW5U 46843042 EC50 = 402 nM T99402 CSUE85 46853657 EC50 = 1100 nM T99402 C1OPF3 46853659 EC50 = 1800 nM T99402 CBZE98 46853681 EC50 = 136 nM T99402 CU9K2H 46853682 EC50 = 179 nM T99402 C0XLK6 46853732 EC50 = 1800 nM T99402 C2RK6A 46853778 EC50 = 6400 nM T99402 CT1W2Q 46869940 EC50 = 99.5 nM T99402 CM24PC 46869941 EC50 = 517 nM T99402 C5F0HL 46869942 EC50 = 556 nM T99402 CEY78X 46869943 EC50 = 6200 nM T99402 C5YV0Z 46869944 EC50 = 41.9 nM T99402 CX1ST9 46869949 EC50 = 435 nM T99402 C1Y0QK 46869950 EC50 = 1400 nM T99402 C8OY4U 46869951 EC50 = 158 nM T99402 C8RL3S 46869952 EC50 = 771 nM T99402 CKB74O 46918013 EC50 = 540 nM T99402 C1VY4Z 46918015 EC50 = 1500 nM T99402 C7KSH2 46918017 EC50 = 8500 nM T99402 CJM4V9 46927956 EC50 > 100000 nM T99402 C01RWE 46934289 EC50 = 19.8 nM T99402 CO3HM4 47131350 IC50 = 5.248 nM T99402 CDWE18 49862462 EC50 > 30000 nM T99402 CE0YN5 49862463 EC50 > 30000 nM T99402 CA4GT5 49862464 EC50 > 30000 nM T99402 C1OE5S 49862522 EC50 = 200 nM T99402 CY7WK6 49862523 EC50 = 1600 nM T99402 CBS63F 49862524 EC50 > 30000 nM T99402 C1XYQ7 49862526 EC50 = 600 nM T99402 C7E6KI 49862527 EC50 = 1600 nM T99402 CAC6F4 49862528 EC50 = 1300 nM T99402 CZQT58 49862579 EC50 = 15800 nM T99402 C9R6BA 49862580 EC50 > 30000 nM T99402 CJ9MI2 49862581 EC50 = 2900 nM T99402 C1YAM2 49862631 EC50 = 4500 nM T99402 COVC28 49862632 EC50 = 4500 nM T99402 CA5TG8 49862633 EC50 > 30000 nM T99402 CDA08M 49862634 EC50 > 30000 nM T99402 CP8S0T 49862635 EC50 > 30000 nM T99402 CF10CB 49862636 EC50 > 30000 nM T99402 CF45MY 49862637 EC50 > 30000 nM T99402 CIB5D2 49862638 EC50 > 30000 nM T99402 CNX34Z 49862693 EC50 = 4100 nM T99402 CY8M4T 49862694 EC50 = 9400 nM T99402 CCO2Y1 49862695 EC50 = 11700 nM T99402 CG9P1F 49862696 EC50 = 16400 nM T99402 CZ0TJ4 49862697 EC50 > 30000 nM T99402 CGM0B2 49862698 EC50 = 5000 nM T99402 CQ83VD 49865230 EC50 = 325 nM T99402 CY91SO 49865291 EC50 > 5000 nM T99402 C5L7JI 49865292 EC50 > 5000 nM T99402 C8S4YA 49865293 EC50 > 10000 nM T99402 C8PMC3 49865350 EC50 = 122 nM T99402 C8SVH2 49865352 EC50 = 478 nM T99402 CC4E6R 49865397 EC50 = 77.4 nM T99402 CI9JM1 49865398 EC50 = 269 nM T99402 CJ94AI 49865399 EC50 = 990 nM T99402 CTK3H1 49865400 EC50 = 686 nM T99402 C15LHQ 49865401 EC50 = 132 nM T99402 CAH15T 49865451 EC50 = 731 nM T99402 CLS5P0 49865452 EC50 = 237 nM T99402 C9PCU5 49865453 EC50 = 2170 nM T99402 CM3TJ5 51003231 EC50 = 627 nM T99402 C8ZV3D 51003232 EC50 = 845 nM T99402 CAJS26 51003233 EC50 = 1780 nM T99402 C6AC2Z 51003234 EC50 = 1330 nM T99402 CUOI26 51003236 EC50 = 1120 nM T99402 CEY7B0 51003281 EC50 = 2090 nM T99402 CZJ5N4 51003282 EC50 = 1605 nM T99402 C1SU4Y 51003283 EC50 = 958 nM T99402 CEY0A6 51003284 EC50 = 426 nM T99402 CCW1T8 51003324 EC50 = 361 nM T99402 C0K8AQ 51003325 EC50 = 114 nM T99402 CF98VG 51003326 EC50 = 4270 nM T99402 CEW46B 51003327 EC50 = 2380 nM T99402 CKRO35 51003329 EC50 = 2150 nM T99402 CTR6J8 51003372 EC50 = 2180 nM T99402 C2L1KF 51003373 EC50 = 403 nM T99402 CU48WB 51003374 EC50 = 1040 nM T99402 C8NTD4 51003375 EC50 = 4720 nM T99402 C0L2SP 51036108 EC50 > 30000 nM T99402 CAU6D5 51036701 EC50 > 30000 nM T99402 CBI3A0 51036916 EC50 > 30000 nM T99402 C3GQ8O 51037131 EC50 > 30000 nM T99402 CE4KP1 51050257 Ki > 10000 nM T99402 CEFL30 51347212 EC50 = 173.78 nM T99402 C86EVA 51352627 EC50 = 110 nM T99402 CFT29A 52913077 EC50 = 398 nM T99402 CNS9J3 52913078 EC50 = 2951.21 nM T99402 C1H3TQ 52913659 EC50 = 104 nM T99402 CX1YO2 52913660 EC50 = 122 nM T99402 C0NMR5 52913766 EC50 = 1230.27 nM T99402 CQJ5F8 52913768 EC50 = 572 nM T99402 CJG3H7 52913772 EC50 = 251 nM T99402 C35JAZ 52913885 EC50 = 190 nM T99402 CP8QC6 52914100 EC50 = 740 nM T99402 C0EXK9 52914105 EC50 = 739 nM T99402 C57CWV 52914203 EC50 = 4168.69 nM T99402 CWE5F0 52914310 EC50 = 84 nM T99402 CT8OX6 52914548 EC50 = 268 nM T99402 C6IEB4 52914664 EC50 = 61.66 nM T99402 CG67LB 52914665 EC50 = 162.18 nM T99402 CN9MF2 52934736 EC50 = 147.91 nM T99402 CV1KU7 52935189 EC50 = 239.88 nM T99402 C8SD6H 52941386 EC50 > 100000 nM T99402 CP97IL 52941387 EC50 > 100000 nM T99402 CN07TX 52944782 EC50 > 100000 nM T99402 CL4EM5 52947232 EC50 > 100000 nM T99402 C8JM1S 52947499 EC50 > 100000 nM T99402 CP8U6O 52948863 EC50 > 100000 nM T99402 CN1HU8 53235518 EC50 > 10000 nM T99402 CY58NO 53240406 EC50 > 25000 nM T99402 C9QI0U 53322767 EC50 = 1410 nM T99402 C04LRU 53324349 EC50 = 1420 nM T99402 CC4BK3 53374105 EC50 = 3590 nM T99402 CLO54R 53375080 EC50 = 67 nM T99402 C8GE6J 53387559 EC50 > 10000 nM T99402 C3XOA8 53387560 EC50 > 10000 nM T99402 C5PWI8 53387561 EC50 = 2200 nM T99402 CO27JT 53387722 EC50 > 10000 nM T99402 CH1WF8 53387723 EC50 > 10000 nM T99402 CED3W5 53387724 EC50 > 10000 nM T99402 CXJT91 53387725 EC50 > 10000 nM T99402 CC0QO6 53387726 EC50 = 1300 nM T99402 C5VJW6 53387727 EC50 > 10000 nM T99402 C9QZV0 53387882 EC50 = 3200 nM T99402 CT8O6H 53387883 EC50 = 2400 nM T99402 CXZ79F 53387884 EC50 > 10000 nM T99402 CPTS36 53387885 EC50 > 10000 nM T99402 C4WFS3 53387886 EC50 = 1300 nM T99402 C6WFI5 53387887 EC50 = 3400 nM T99402 CI18AF 53388040 EC50 > 10000 nM T99402 CMI7W4 53388041 EC50 > 10000 nM T99402 C46FKH 53388042 EC50 = 290 nM T99402 C3K7OI 53388191 EC50 = 4900 nM T99402 CA9BN5 53388192 EC50 > 10000 nM T99402 CT1P5F 53388193 EC50 = 2700 nM T99402 C5AZ0O 53388194 EC50 = 390 nM T99402 CXF6A5 53388195 EC50 = 340 nM T99402 C5G1NQ 53388196 EC50 = 600 nM T99402 CJD0H2 53388197 EC50 > 10000 nM T99402 CWO0G6 53388362 EC50 = 100 nM T99402 CA38RS 53495171 EC50 = 83 nM T99402 CIHC67 54582001 IC50 > 30000 nM T99402 CDZX39 54670123 EC50 = 446.68 nM T99402 CYV78T 54670222 EC50 = 4137 nM T99402 CP58ID 54670223 EC50 = 547 nM T99402 CE76FW 54670224 EC50 = 295 nM T99402 C52ZCU 54670496 EC50 = 217 nM T99402 C4GH7A 54670499 EC50 = 150 nM T99402 CR87TD 54670965 EC50 = 189 nM T99402 CJRG27 54761054 EC50 > 30000 nM T99402 CT73PK 54764842 IC50 = 8200 nM T99402 C2IO3D 56649042 EC50 = 353 nM T99402 C1YVN5 56649043 EC50 = 104 nM T99402 CJ4RU3 57391480 IC50 = 7700 nM T99402 C6RK0U 57391482 IC50 > 10000 nM T99402 C4MFY7 57391520 EC50 = 4600 nM T99402 CE9X1S 57393242 IC50 > 10000 nM T99402 CL5M4D 57393245 IC50 = 4700 nM T99402 CL1KN7 57393246 IC50 > 10000 nM T99402 C6W1FB 57396719 IC50 = 8000 nM T99402 CO9F2S 57396720 IC50 > 10000 nM T99402 C6W7LD 57478075 EC50 = 2700 nM T99402 CZ0A1T 57765525 EC50 = 2800 nM T99402 CE7DU0 57765529 EC50 = 1500 nM T99402 C6N0PK 57765531 EC50 = 1600 nM T99402 C49IAZ 57765535 EC50 = 2000 nM T99402 C4BZ0U 57765536 EC50 = 380 nM T99402 C9QDZ0 57765549 EC50 = 241000 nM T99402 C90MQS 57765556 EC50 = 2400 nM T99402 CHQM83 57765572 EC50 = 1600 nM T99402 C4T6JE 57765594 EC50 = 900 nM T99402 C1K5DT 57765607 EC50 = 23000 nM T99402 CSI9E0 57765613 EC50 = 440 nM T99402 CZ4KT6 57765615 EC50 = 1760 nM T99402 CBFD61 57765616 EC50 = 400 nM T99402 CC82HD 57765622 EC50 = 380 nM T99402 CQ70WE 57765633 EC50 = 490 nM T99402 CISA81 58058356 EC50 = 4300 nM T99402 CPDW56 58058372 EC50 = 420 nM T99402 CQY10C 58058380 EC50 = 11600 nM T99402 CY2NR8 58058384 EC50 = 540 nM T99402 C8N4UB 60096231 EC50 = 11757 nM T99402 C3HZ5J 60150507 EC50 = 220 nM T99402 CZB79F 62316492 IC50 = 7.4 nM T99402 C4PU9N 67056056 EC50 > 30000 nM T99402 CBX67G 67246999 EC50 > 10000 nM T99402 C5K7QG 67974411 EC50 > 10000 nM T99402 C0BC6D 68012045 EC50 = 19000 nM T99402 CCT07V 68290289 EC50 > 10000 nM T99402 C03JUE 68290572 EC50 > 10000 nM T99402 C13MPG 68374199 EC50 = 1021 nM T99402 CPL87R 68374351 EC50 = 344 nM T99402 CZT05A 69929646 EC50 > 30000 nM T99402 CZ0TQ4 70681379 EC50 = 3100 nM T99402 CG63WO 70681380 EC50 = 4300 nM T99402 CW4D7F 70683514 EC50 > 10000 nM T99402 C3K8DF 70683515 EC50 = 2800 nM T99402 CSEH49 70683516 EC50 > 10000 nM T99402 C1L9YU 70683517 EC50 = 1800 nM T99402 CNSH92 70683518 EC50 = 690 nM T99402 CRC38L 70683529 EC50 = 950 nM T99402 C5S6IR 70683530 EC50 = 10000 nM T99402 COF23E 70683531 EC50 = 2400 nM T99402 C50OCJ 70683532 EC50 = 1200 nM T99402 CV43BW 70685621 EC50 > 10000 nM T99402 CU50QS 70687762 EC50 = 480 nM T99402 CFK1R6 70687763 EC50 = 590 nM T99402 CKH1F4 70687764 EC50 = 640 nM T99402 C2BPE5 70687765 EC50 = 250 nM T99402 C31UQX 70687777 EC50 = 2500 nM T99402 CB36GD 70687778 EC50 = 5100 nM T99402 C0EQ4T 70689779 EC50 = 2100 nM T99402 CB0HM2 70689815 EC50 = 730 nM T99402 CMNK78 70689822 EC50 = 390 nM T99402 C1U6CJ 70691951 EC50 = 540 nM T99402 CN4WZ1 70691952 EC50 > 10000 nM T99402 CB76TW 70691953 EC50 > 10000 nM T99402 CJ3R7H 70691954 EC50 = 6000 nM T99402 CX9BH7 70691970 EC50 = 190 nM T99402 CS9RX5 70691971 EC50 = 3500 nM T99402 CTN61K 70691972 EC50 = 2300 nM T99402 CBT84P 70693972 EC50 = 1100 nM T99402 CDUO86 70694002 EC50 = 670 nM T99402 CAR57I 70694003 EC50 = 550 nM T99402 CC27HR 70694004 EC50 = 390 nM T99402 CU2C9B 70694005 EC50 > 10000 nM T99402 CK85GB 70696128 EC50 = 840 nM T99402 CDL51A 70696130 EC50 > 10000 nM T99402 C58ELH 70696137 EC50 = 500 nM T99402 C3F4HT 70696138 EC50 = 900 nM T99402 CC6AS8 71260327 EC50 = 188 nM T99402 CNIW83 71479388 EC50 > 30000 nM T99402 CXW8R2 72714783 EC50 > 10000 nM T99402 C7ORB6 73058507 EC50 = 108 nM T99402 CHS04F 87304250 EC50 = 1710 nM T99402 C3G0XF 87304273 EC50 = 2340 nM T99402 CX5BE2 87305070 EC50 = 46 nM T99402 C07OAB 87618914 EC50 = 1400 nM T99402 C7DP6O 88957119 EC50 = 436.52 nM T99402 CZ23DK 89106981 EC50 = 165 nM T99402 C4Q7OH 89115789 EC50 = 160 nM T99402 CH4L7O 91885483 EC50 > 10000 nM T99402 C0VN8X 92044496 EC50 = 160 nM T99402 CIF0U7 113447561 EC50 = 575.44 nM T99402 CF84JO 113943306 IC50 = 7.3 nM T99402 C2T1FS 115497227 IC50 = 6.607 nM T99402 CJ5G3Q 118718091 EC50 > 1000000 nM T99402 C2IA6C 121485534 EC50 = 269 nM T99402 C7K8UR 121485558 EC50 = 794 nM T99402 CR21EM 121485560 EC50 = 1047.13 nM T99402 CMUP23 122187789 EC50 = 291 nM T99402 CP7R1A 122187790 IC50 = 322 nM T99402 C74XFR 122187791 IC50 = 144.54 nM T99402 CAQ0N6 122187792 IC50 = 47 nM T99402 C23JFU 122187793 IC50 = 169.82 nM T99402 C72YXV 122187794 IC50 = 3.2 nM T99402 CUC13P 122187795 IC50 = 3.236 nM T99402 CJV7O0 122187796 IC50 = 3.7 nM T99402 CMHP48 122193173 EC50 = 616.6 nM T99402 CE1L3P 122193174 EC50 = 323 nM T99402 CJIB74 122193175 EC50 = 1140 nM T99402 C1N0HP 122193176 EC50 = 2250 nM T99402 CV8J6N 122193177 EC50 = 1110 nM T99402 C01PDA 122193178 EC50 = 712 nM T99402 CB8MH7 122193179 EC50 < 10000 nM T99402 CCP5U2 122195692 EC50 > 10000 nM T99402 CWHE41 122196091 EC50 > 10000 nM T99402 CEG8I0 122196092 EC50 = 350 nM T99402 C2KA8E 122196093 EC50 = 483 nM T99402 C6TI1L 122196094 EC50 = 382 nM T99402 COC02R 122196095 EC50 = 265 nM T99402 CO48MD 122196096 EC50 = 287 nM T99402 CR34BM 122196097 EC50 = 264 nM T99402 CMUE28 122196098 EC50 = 674 nM T99402 C9WU0F 122196099 EC50 = 885 nM T99402 C2FI9X 122196100 EC50 = 422 nM T99402 C0BK2L 122196101 EC50 = 1010 nM T99402 CS42ED 122196102 EC50 = 1100 nM T99402 CPE1I5 122196103 EC50 = 6660 nM T99402 CVIB23 122196104 EC50 = 5760 nM T99402 CK2Z0Y 122196105 EC50 = 2470 nM T99402 C5ODB4 122196106 EC50 = 2870 nM T99402 CER92P 122196107 EC50 = 1180 nM T99402 C4W6FN 122196108 EC50 = 882 nM T99402 C91DKH 122196109 EC50 = 647 nM T99402 CVFI45 122196110 EC50 = 1930 nM T99402 CK6Q3M 122196111 EC50 > 10000 nM T99402 CB7FN6 122196112 EC50 = 5000 nM T99402 CZ08OD 122196113 EC50 = 1113 nM T99402 C4VWT9 122196114 EC50 = 3550 nM T99402 C65ABR 122196115 EC50 = 4670 nM T99402 CY9PM2 122196116 EC50 = 4470 nM T99402 CRB9G8 122196117 EC50 = 2530 nM T99402 CU7JC9 122196118 EC50 > 10000 nM T99402 CHT0B7 122196119 EC50 = 353 nM T99402 CZ0HS9 122196120 EC50 = 429 nM T99402 C7LP8W 122196121 EC50 = 513 nM T99402 CG5O4N 122196122 EC50 = 809 nM T99402 C2EXU4 122196123 EC50 > 10000 nM T99402 CZ94FU 122196124 EC50 > 10000 nM T99402 CM6T9O 122196125 EC50 = 609 nM T99402 CF8CV6 122196126 EC50 > 10000 nM T99402 C7PA4V 122196127 EC50 > 10000 nM T99402 C2MK3Z 122196128 EC50 > 10000 nM T99402 CEV41Y 122196129 EC50 > 10000 nM T99402 CB2N5C 122419056 EC50 = 81 nM T99402 CLRU07 122419058 EC50 = 67.61 nM T99402 CG60YJ 122419061 EC50 = 104.71 nM T99402 C91EHA 122419063 EC50 = 199.53 nM T99402 C1BUR9 122419071 EC50 = 758.58 nM T99402 CBCI87 122419072 EC50 = 323.59 nM T99402 CIP79O 122419073 EC50 = 81 nM T99402 C7XH6S 122419077 EC50 = 26 nM T99402 CL4CX1 122419141 EC50 = 398 nM T99402 C8C7RT 122419143 EC50 = 446.68 nM T99402 CD1J0S 122419145 EC50 = 67.61 nM T99402 CW61PJ 122419153 EC50 = 389 nM T99402 C7GA2E 122419157 EC50 = 331 nM T99402 CGT12J 122419159 EC50 = 50.1 nM T99402 CERA43 122419160 EC50 = 323.59 nM T99402 C5-NOV-09 122419161 EC50 = 275 nM T99402 C3PAN4 122419163 EC50 = 52.4 nM T99402 CH2AO4 122539788 IC50 > 30000 nM T99402 C2MEI0 124425164 EC50 = 4400 nM T99402 C2K9ZI 127025479 EC50 = 1120 nM T99402 C2XF0N 127025548 EC50 = 198 nM T99402 CIX4C9 127025549 EC50 = 519 nM T99402 CM56OW 127025550 EC50 = 983 nM T99402 CX57FG 127025563 EC50 = 474 nM T99402 C7TVF2 127025564 EC50 = 602 nM T99402 CGYD41 127025831 EC50 = 642 nM T99402 CY9ZE6 127025845 EC50 = 506 nM T99402 CH78CV 127025846 EC50 > 10000 nM T99402 CSXW80 127025847 EC50 = 1070 nM T99402 C7FQ0Z 127025860 EC50 > 10000 nM T99402 CECS36 127025861 EC50 > 10000 nM T99402 C47QGK 127026059 EC50 > 10000 nM T99402 CDJ6A7 127026067 EC50 = 1410 nM T99402 C0S2UW 127026137 EC50 = 2530 nM T99402 C1G5PU 127026138 EC50 = 1980 nM T99402 CV3I2A 127026139 EC50 > 10000 nM T99402 CPB15M 127026140 EC50 = 306 nM T99402 CQ09MN 127026386 EC50 > 10000 nM T99402 CFNI82 127026469 EC50 = 1090 nM T99402 CG8L6K 127026470 EC50 > 10000 nM T99402 CHJ2V0 127026471 EC50 = 2750 nM T99402 CJH69G 127026472 EC50 = 3380 nM T99402 C03DLS 127026473 EC50 > 10000 nM T99402 C82JTZ 127026474 EC50 = 6200 nM T99402 CEDC20 127028298 EC50 = 1573 nM T99402 CGJ86U 127028301 EC50 > 10000 nM T99402 C3SDP4 127028303 EC50 = 405 nM T99402 C2POU1 127033963 EC50 > 10000 nM T99402 C8Q6BJ 127043558 EC50 = 5000 nM T99402 C8YG3A 127044238 EC50 > 30000 nM T99402 C81XER 127046201 EC50 = 3.96 nM T99402 CI8JY9 127046202 EC50 > 10 nM T99402 C3XQ4S 127046203 EC50 = 1.25 nM T99402 CORL35 127046204 EC50 > 10 nM T99402 CIS24M 127046205 EC50 > 10 nM T99402 C4TY6B 127046254 EC50 = 2.52 nM T99402 C9A1TG 127046557 EC50 = 0.095 nM T99402 C4D3ST 127046558 EC50 = 0.689 nM T99402 CW39BI 127046775 EC50 = 0.236 nM T99402 CRH43X 127046929 EC50 > 10 nM T99402 C14UHR 127046933 EC50 = 2.8 nM T99402 C4WF1O 127046934 EC50 = 1.86 nM T99402 C4O7GW 127046935 EC50 = 1.28 nM T99402 CM6W3S 127047061 EC50 = 0.758 nM T99402 CCQ3S2 127047065 EC50 = 0.921 nM T99402 CU10TY 127047066 EC50 > 10 nM T99402 CKT86B 127047343 EC50 = 1.61 nM T99402 C49CXE 127047638 EC50 = 2.19 nM T99402 C7YML2 127047647 EC50 = 0.065 nM T99402 COH3C7 127047648 EC50 = 1.35 nM T99402 CF9K6R 127047649 EC50 = 125 nM T99402 CL2QM3 127047650 EC50 > 10000 nM T99402 CY3R6Q 127047763 EC50 = 296 nM T99402 C1G8VO 127048133 EC50 = 0.319 nM T99402 CPZ70S 127052897 EC50 > 30000 nM T99402 C38BRY 131801162 EC50 > 10000 nM T99402 CFC05Q 131954513 EC50 > 10000 nM T99402 C9WH5Q 134189963 EC50 = 723 nM T99402 CBP6O9 134189964 EC50 = 1348.96 nM T99402 C2N8ZW 134189970 EC50 = 812.83 nM T99402 CG04WB 134189978 EC50 = 512.86 nM T99402 CM4F0T 134189979 EC50 = 707.95 nM T99402 C72PMB 134189980 EC50 = 851 nM T99402 C7NR1Y 134189992 EC50 = 1288.25 nM T99402 C6V3NP 134189994 EC50 = 1860 nM T99402 CU6TG2 134190027 EC50 = 851.14 nM T99402 C8LV4C 134190028 EC50 = 2818.38 nM T99402 C8O3WA 134190146 EC50 = 676.08 nM T99402 CZ13MP 134190171 EC50 = 2398.83 nM T99402 C71ZAO 134190172 EC50 = 75.86 nM T99402 C0RTE8 134190173 EC50 = 227 nM T99402 C5E8TU 134190176 EC50 = 137 nM T99402 CLE08W 134190209 EC50 = 524.81 nM T99402 CWSD56 134190210 EC50 = 128.82 nM T99402 CPR9G4 134190211 EC50 = 97.72 nM T99402 C4K2VM 134190218 EC50 = 117 nM T99402 CJP62Y 134190222 EC50 = 1570 nM T99402 CU8O6H 134190223 EC50 = 218.78 nM T99402 C8F6EB 134190224 EC50 = 22.9 nM T99402 CL5PJ6 134190225 EC50 = 122 nM T99402 C0IFS2 134190227 EC50 = 274 nM T99402 CG31VY 134190246 EC50 = 575 nM T99402 CVFK58 134191934 EC50 = 43 nM T99402 CYM7D1 134191937 EC50 = 19.8 nM T99402 CH2S0D 134191938 EC50 = 43.2 nM T99402 C89OZT 134191951 EC50 = 67.9 nM T99402 C7MBI1 134191954 EC50 = 78.1 nM T99402 C7SOG4 134191958 EC50 = 129 nM T99402 CEK67R 134191960 EC50 = 37.9 nM T99402 CP9H5A 134191963 EC50 = 24.9 nM T99402 CHR7V0 134191965 EC50 = 413 nM T99402 C95VMR 134191976 EC50 = 104 nM T99402 CSYW09 134191981 EC50 = 95.1 nM T99402 C27YHQ 134192002 EC50 = 1880 nM T99402 CVH6K5 134192017 EC50 = 468 nM T99402 CJX1D4 134192043 EC50 = 452 nM T99402 CX39GM 134192044 EC50 = 1210 nM T99402 C0TDN1 134192062 EC50 = 231 nM T99402 C78NTY 134192068 EC50 = 9890 nM T99402 COM29G 134192169 EC50 = 45.4 nM T99402 CTI5Q4 134198051 EC50 = 85.6 nM T99402 C7BMY9 134198072 EC50 = 827 nM T99402 CTW92Y 134198074 EC50 = 653 nM T99402 C4Y2PO 134198076 EC50 = 289 nM T99402 CHF54I 134198077 EC50 = 345 nM T99402 CU01QM 134198078 EC50 = 794 nM T99402 CKX61P 134198081 EC50 = 764 nM T99402 CR4SL5 134198083 EC50 = 116 nM T99402 CBSU83 134198103 EC50 = 815 nM T99402 CRTP47 134198221 EC50 = 46.8 nM T99402 C9IKH0 134198340 EC50 = 265 nM T99402 CVN95I 134198344 EC50 = 498 nM T99402 CC13EJ 134198363 EC50 = 870 nM T99402 C8JIS7 135125589 EC50 = 1269 nM T99402 CV8IE5 135125797 EC50 = 2509 nM T99402 CM05YJ 135125800 EC50 = 1320 nM T99402 CDH3C9 135125802 EC50 = 464 nM T99402 CFG70D 135125807 EC50 = 304 nM T99402 C5C1SR 135125813 EC50 = 373 nM T99402 C73WMI 135125821 EC50 = 1031 nM T99402 C5RPE8 135126257 EC50 = 668 nM T99402 CWY06X 135126260 EC50 = 1460 nM T99402 C7U0FS 135126261 EC50 = 3363 nM T99402 CADP15 135126262 EC50 = 648 nM T99402 C5X6DK 135126267 EC50 = 3204 nM T99402 C6XY7H 135126270 EC50 = 952 nM T99402 CJ2V9X 135126274 EC50 = 2631 nM T99402 C08JBT 135126302 EC50 = 1216 nM T99402 CX8AP2 135126561 EC50 > 10000 nM T99402 C4VQ2E 135126567 EC50 = 1388 nM T99402 C8Y4RM 135126573 EC50 = 116 nM T99402 CF0Y4Z 135126574 EC50 = 737 nM T99402 CJZ24Q 135998881 EC50 > 30000 nM T99402 CEQ67U 136254191 EC50 > 10000 nM T99402 CIL04G 136353157 EC50 = 5260 nM T99402 C4FIK0 136415539 EC50 = 90 nM T99402 CW6PU0 136415548 EC50 = 9840 nM T99402 CTO85Q 136415554 EC50 = 35 nM T99402 C2OPU0 136503347 EC50 = 310 nM T99402 C89HFS 136503356 EC50 = 200 nM T99402 CFAY85 136503359 EC50 = 1630 nM T99402 CGBA35 136503360 EC50 = 1720 nM T99402 CV6T4B 136503361 EC50 = 1740 nM T99402 CE54RA 136503365 EC50 = 690 nM T99402 CY37GV 136503366 EC50 = 750 nM T99402 CI85DP 136503369 EC50 = 1160 nM T99402 CD7C3L 136503370 EC50 = 3010 nM T99402 CRWA31 136503371 EC50 = 1270 nM T99402 C4KX9H 136503374 EC50 = 860 nM T99402 C8Y4VJ 136503375 EC50 = 2470 nM T99402 CIF1O4 136503384 EC50 = 240 nM T99402 CU56JI 136503386 EC50 = 130 nM T99402 C3EGM5 137321168 IC50 > 10000 nM T99402 C7PU2H 137631652 EC50 > 30000 nM T99402 C0M7EV 137631886 EC50 = 28000 nM T99402 CMSP48 137631939 EC50 = 50 nM T99402 CH29EQ 137631968 EC50 = 60 nM T99402 CI4V1F 137631983 EC50 = 7800 nM T99402 C8QU9Z 137632643 EC50 = 6400 nM T99402 CP36EU 137633977 EC50 = 980 nM T99402 C4E7KH 137634091 EC50 = 7700 nM T99402 C2WJ3T 137634489 EC50 = 25300 nM T99402 CS7O0A 137634883 EC50 = 2000 nM T99402 CVTW69 137635028 EC50 = 53 nM T99402 CQ02YR 137635378 EC50 = 3400 nM T99402 CTG5M8 137635566 EC50 = 25000 nM T99402 CU2JA5 137636549 EC50 = 33000 nM T99402 C6OVJ8 137637239 EC50 = 3960 nM T99402 C0KAJ3 137638200 EC50 = 6100 nM T99402 C9A8MG 137638288 EC50 = 5100 nM T99402 C5O4LT 137639171 EC50 = 50 nM T99402 C9H6NY 137639752 EC50 = 500 nM T99402 CEG8C1 137639864 EC50 = 4 nM T99402 CK2W6L 137640190 EC50 = 1000 nM T99402 CBVM98 137641505 EC50 = 1390 nM T99402 C7KT0R 137642290 EC50 = 2300 nM T99402 C65YBA 137642559 EC50 = 280 nM T99402 CAI63F 137642874 EC50 = 320 nM T99402 CJHL32 137643079 EC50 = 41000 nM T99402 CNY07D 137643617 EC50 = 4410 nM T99402 C1FCY7 137643759 EC50 = 8800 nM T99402 CS5F0B 137644345 EC50 = 6500 nM T99402 CS7FM3 137644474 EC50 = 17 nM T99402 C0B5SL 137645909 EC50 = 1010 nM T99402 C9U6EI 137645989 EC50 = 720 nM T99402 CCW58E 137646034 EC50 = 24000 nM T99402 C9FAO3 137646208 EC50 = 53 nM T99402 C3PDO0 137647077 EC50 = 1700 nM T99402 C3IFR5 137647687 EC50 = 10 nM T99402 C2AM0L 137648363 EC50 = 6990 nM T99402 CCGJ82 137648591 EC50 = 106 nM T99402 CEBV64 137649482 EC50 = 800 nM T99402 CUH06J 137649749 EC50 = 2000 nM T99402 CO9L1G 137650519 EC50 = 1950 nM T99402 CQKZ08 137651515 EC50 = 15800 nM T99402 CYK1P7 137651881 EC50 = 42000 nM T99402 C6CW1G 137652072 EC50 = 30000 nM T99402 CH5WQ1 137652776 EC50 = 19 nM T99402 C5B0YD 137653133 EC50 = 14210 nM T99402 CT1M7B 137654697 EC50 = 4500 nM T99402 CMQ61F 137655963 EC50 = 9770 nM T99402 CL73HA 137656701 EC50 = 6 nM T99402 CGCT53 137658747 EC50 = 150 nM T99402 C5OK1E 137659207 EC50 = 7900 nM T99402 C46DSV 137659319 EC50 = 25 nM T99402 CDV5F8 137660178 EC50 = 4 nM T99402 CDWR37 137661492 EC50 = 15000 nM T99402 C9C8KU 137661528 EC50 = 2420 nM T99402 CL3GA9 137661688 EC50 = 35 nM T99402 COH64G 140838160 EC50 = 907 nM T99402 CWA8H2 145955288 EC50 > 10000 nM T99402 C7XLW1 145957424 EC50 = 2100 nM T99402 C93IJD 145957567 EC50 > 30000 nM T99402 CQ2TN4 145962919 EC50 > 30000 nM T99402 C6CBO4 145982965 EC50 = 1430 nM T99402 CC6DT0 145983157 EC50 > 10000 nM T99402 CR7W8H 145983574 EC50 = 119 nM T99402 C8ZGU9 145984231 EC50 = 36.2 nM T99402 C1LW9O 145985523 EC50 = 95.5 nM T99402 C9YZ1M 145985934 EC50 = 160 nM T99402 CRM28X 145986132 EC50 = 257 nM T99402 C76FVC 155518354 EC50 = 2100 nM T99402 CYXE53 155538270 IC50 > 10000 nM T99402 CMKT08 155540610 EC50 > 10000 nM T99402 CHD6N7 155549892 EC50 = 39.81 nM T99402 CQ71TD 155557230 EC50 = 74 nM T99402 CYV4P0 155564012 EC50 = 102 nM T99402 D00EPM 73755217 IC50 > 30000 nM T99402 D00IGI 2207 EC50 = 330 nM T99402 D00NCL 46836562 EC50 = 9 nM T99402 D01EVA 6278000 Ki > 100000 nM T99402 D01JFF 44191096 IC50 = 5.1 nM T99402 D01YEN 1233 Ki > 1000000 nM T99402 D03MEI 3260619 EC50 = 4600 nM T99402 D03PGL 46911068 EC50 = 1000 nM T99402 D03UIR 24905704 EC50 > 100000 nM T99402 D04DKM 104766 EC50 = 39000 nM T99402 D04JKL 2071 Ki > 1000000 nM T99402 D04MVR 11530404 IC50 > 10000 nM T99402 D05GQH 46836872 EC50 = 4 nM T99402 D05TFE 5218788 Ki > 100000 nM T99402 D06DUE 40539 Ki = 112000 nM T99402 D06PAK 10058694 Ki > 100000 nM T99402 D07GRG 10197984 Ki = 21000 nM T99402 D07IOB 4052597 EC50 = 3000 nM T99402 D07PZQ 68841 EC50 = 1000 nM T99402 D09AQK 4545574 EC50 = 3200 nM T99402 D09QUN 58368068 EC50 > 10000 nM T99402 D09RPR 16737207 Ki > 10000 nM T99402 D09UBS 10428048 Ki > 100000 nM T99402 D0EK6P 5310984 Ki > 300000 nM T99402 D0IO8J 3025961 Ki > 100000 nM T99402 D0J2WN 5311344 Ki = 50000 nM T99402 D0K2XD 53391766 IC50 > 10000 nM T99402 D0KL4K 71041983 EC50 = 110 nM T99402 D0L0YF 4236420 EC50 > 3000000 nM T99402 D0LC5O 16062593 EC50 = 1960 nM T99402 D0N0NJ 15508178 IC50 > 300000 nM T99402 D0N2TP 44190040 IC50 > 10000 nM T99402 D0N9UZ 9819927 Ki = 22000 nM T99402 D0OH2P 5311040 Ki > 300000 nM T99402 D0OV2V 6324634 Ki > 300000 nM T99402 D0P3XO 5311459 Ki = 838000 nM T99402 D0PN6Z 179394 EC50 = 100 nM T99402 D0Q6VH 5311432 Ki = 26000 nM T99402 D0T5SU 158397 EC50 > 3000000 nM T99402 D0V8KA 42645487 EC50 = 410 nM T99402 D0W3PY 6604820 EC50 = 1700 nM T99402 D0W9VN 836002 EC50 = 1100 nM T99402 D0X3VM 888023 EC50 = 740 nM T99402 D0YO8B 5311457 Ki > 1000000 nM T99402 D0Z5JT 135773804 EC50 = 1700 nM T62450 CCXJ65 462474 IC50 = 1200 nM T62450 C5WH9E 462475 IC50 = 780 nM T62450 C1G0QS 462476 IC50 = 110 nM T62450 C24KOA 469465 IC50 = 16000 nM T62450 CR90KX 469467 IC50 = 19000 nM T62450 C89ZBY 469469 IC50 = 8200 nM T62450 C9MGQ5 469470 IC50 = 360 nM T62450 CW06GL 469471 IC50 = 760 nM T62450 C49UAY 469473 IC50 = 600 nM T62450 C7PZ2G 469475 IC50 = 300 nM T62450 C7O3GY 469477 IC50 = 5200 nM T62450 CFD9R0 469479 IC50 > 100000 nM T62450 CF69BX 469481 IC50 = 270 nM T62450 CM7TQ8 469483 IC50 = 350 nM T62450 CO92AX 469485 IC50 = 690 nM T62450 C62NEY 469486 IC50 = 6700 nM T62450 CN1L7J 469488 IC50 > 10000 nM T62450 CZ7FD4 469490 IC50 = 1200 nM T62450 CQ1IT6 469492 IC50 = 5000 nM T62450 CWD38H 469494 IC50 = 1300 nM T62450 CUW1Y2 469495 IC50 = 190 nM T62450 C18AYG 469497 IC50 = 110 nM T62450 CKL4D6 469498 IC50 = 750 nM T62450 CF3DJ4 469499 IC50 = 520 nM T62450 C9R0JO 469500 IC50 = 170 nM T62450 CA80IT 469501 IC50 = 340 nM T62450 C8BN6K 469502 IC50 > 10000 nM T62450 COA3R4 469503 IC50 = 750 nM T62450 CG09VN 469504 IC50 = 43 nM T62450 CRI0U5 469579 IC50 = 365000 nM T62450 CNWM94 489104 IC50 = 980 nM T62450 CX6LW0 489106 IC50 = 1200 nM T62450 C6WKB1 489107 IC50 = 1700 nM T62450 CW46FX 489108 IC50 = 50000 nM T62450 CFC9M3 489109 IC50 = 4400 nM T62450 CK9C8M 489110 IC50 = 1500 nM T62450 CP18RH 489111 IC50 = 1600 nM T62450 C2VFD3 491343 IC50 = 620 nM T62450 C0PSK1 491351 IC50 = 5.7 nM T62450 C35LZD 500952 IC50 = 0.39 nM T62450 CKW8G7 5274768 IC50 = 34 nM T62450 C23VBK 5274769 IC50 = 110 nM T62450 COJ3M2 5274770 IC50 = 74 nM T62450 CS3B7G 5274771 IC50 = 300 nM T62450 CMG84V 5274772 IC50 = 65 nM T62450 CD82HT 5274773 IC50 = 190 nM T62450 CC0BF4 5274774 IC50 = 500 nM T62450 CSMQ62 5274775 IC50 = 26 nM T62450 CZL93E 5274776 IC50 = 210 nM T62450 CFK94B 5274777 IC50 > 10000 nM T62450 C6XNB3 5274778 IC50 = 1900 nM T62450 C7AJ8N 5274779 IC50 = 2300 nM T62450 CXKI49 5274787 IC50 > 10000 nM T62450 CMU5J6 5274788 IC50 > 10000 nM T62450 CON32R 5274789 IC50 > 10000 nM T62450 CI4OB1 5274790 IC50 > 10000 nM T62450 C41DUG 5274791 IC50 > 1000 nM T62450 CKC79R 5274792 IC50 > 10000 nM T62450 C02UYM 5274793 IC50 > 10000 nM T62450 CPN1U4 5274794 IC50 = 130 nM T62450 COCT-69 5274795 IC50 = 46 nM T62450 COI21Y 5274796 IC50 = 28 nM T62450 CG28JL 5274797 IC50 = 23 nM T62450 CU9EM1 5274798 IC50 = 890 nM T62450 C1G5PL 5274800 IC50 = 160 nM T62450 C0B8HY 5274801 IC50 > 10000 nM T62450 C6I7PW 5274802 IC50 > 10000 nM T62450 C9J7ZL 5274803 IC50 = 730 nM T62450 CF8N7V 5274804 IC50 > 10000 nM T62450 C4ZDE6 5274805 IC50 > 10000 nM T62450 CLM8B1 5274806 IC50 > 10000 nM T62450 C3JT2S 5274807 IC50 = 310 nM T62450 CU1R7E 5274808 IC50 = 160 nM T62450 CN2SM9 5274811 IC50 = 11 nM T62450 CA65PW 5274815 IC50 = 0.49 nM T62450 C0E7FP 5276704 IC50 = 0.49 nM T62450 CV0J6T 5481068 IC50 = 16000 nM T62450 C13DPV 9873540 IC50 = 20000 nM T62450 CRF91L 10393588 IC50 = 29300 nM T62450 C5JWZ8 10483511 IC50 = 17500 nM T62450 C62JDA 10531055 IC50 = 300 nM T62450 CO0CG6 10816011 IC50 = 3900 nM T62450 CZ5O8K 11455046 IC50 = 2.3 nM T62450 COQ1M3 44445039 IC50 > 10000 nM T62450 C7CNE6 44445040 IC50 = 15 nM T62450 CP7CI1 44445043 IC50 = 130 nM T62450 C3M9UG 44445044 IC50 = 3.3 nM T62450 C81XCA 44445045 IC50 = 2.4 nM T62450 CKI5L4 44445048 IC50 = 8.1 nM T62450 C1DCS7 44445049 IC50 = 34 nM T62450 CTO09N 76308527 IC50 = 10000 nM T62450 CV9X8D 76312215 IC50 = 1200 nM T62450 CIH2U1 76315758 IC50 = 620 nM T62450 C9KRV6 76315759 IC50 = 83000 nM T62450 C2BS9Y 76315760 IC50 = 3.7 nM T62450 C89MVI 76315761 IC50 = 7.5 nM T62450 C02NVW 76319451 IC50 = 454569193.6 nM T62450 CD93UK 76319452 IC50 = 3 nM T62450 CZ68WH 76319453 IC50 = 17001999.54 nM T62450 C7YRE5 76319454 IC50 = 72011192.02 nM T62450 C73UVY 76319455 IC50 = 8.3 nM T62450 CV6E1G 76319456 IC50 = 5201157.44 nM T62450 CP9N0A 76323072 IC50 = 3300 nM T62450 C3VBU9 76323073 IC50 = 1 nM T62450 CG6AW9 76323074 IC50 = 9401561.69 nM T62450 C4BKS3 76326640 IC50 = 4400 nM T62450 C8RI0A 76326641 IC50 = 100 nM T62450 CP82OB 76326642 IC50 = 79000 nM T62450 CE2C7R 76326643 IC50 = 73 nM T62450 CB85FY 76330302 IC50 = 110001852.8 nM T62450 C7D3LY 76330303 IC50 = 5.7 nM T62450 CO0NB3 118718710 IC50 = 80000 nM T62450 C7AOF2 118718711 IC50 = 110000 nM T84173 D03DSR 2132 IC50 = 4100 nM T84173 D0D0ZD 441314 IC50 = 84000 nM T84173 D0HR8Z 51634 IC50 = 118000 nM T84173 D0RE9C 501391 IC50 = 320000 nM T84173 D0S5LT 29435 Ki = 2000 nM T84173 CF4VT6 61163 Ki = 620000 nM T84173 C65JPY 68215 IC50 > 500000 nM T84173 CEIH96 75059 IC50 > 500000 nM T84173 C6P0QT 129374 IC50 = 500000 nM T84173 CXH6Y5 183073 Ki = 6300 nM T84173 CML92R 272783 IC50 > 500000 nM T84173 C2A6JZ 348641 IC50 > 500000 nM T84173 CHY93K 447607 IC50 = 59 nM T84173 C1EH0P 501640 Ki = 300 nM T84173 C4NG2D 650378 Ki = 320 nM T84173 C7UG5A 762600 IC50 > 500000 nM T84173 CO7VU1 787204 IC50 > 500000 nM T84173 CROP13 873720 IC50 = 177 nM T84173 C6QBR5 874599 IC50 = 97 nM T84173 CQI01W 1241968 Ki = 50600 nM T84173 C1VXR6 1300581 Ki = 102 nM T84173 CV20DJ 1309961 IC50 = 2960 nM T84173 C5JK1V 1310191 Ki = 19200 nM T84173 C2PEY8 1362627 IC50 = 6460 nM T84173 CAQ2S5 2055451 Ki = 4230 nM T84173 CD7V1H 2210290 Ki = 52 nM T84173 CBX4C0 2224401 Ki = 7150 nM T84173 C1BDJ3 2456688 IC50 = 42 nM T84173 CV1NZ9 3141863 IC50 = 47700 nM T84173 C7Q1XB 3141864 IC50 = 46500 nM T84173 CD7HS0 3146158 Ki = 2780 nM T84173 C2ZR5W 3146886 IC50 = 12130 nM T84173 CBU70S 3237927 Ki = 56 nM T84173 CH9TY7 3262578 Ki = 2500 nM T84173 C4SPY2 3448473 IC50 > 500000 nM T84173 CV2Z4B 4244680 Ki = 975 nM T84173 CI4LF2 4767568 IC50 = 16470 nM T84173 C6ITG1 4882879 IC50 = 36070 nM T84173 CL45KY 4965949 IC50 = 20 nM T84173 CV8C9W 5067281 Ki = 21 nM T84173 CD03RL 7663529 IC50 > 500000 nM T84173 CPJX49 8080175 IC50 = 28070 nM T84173 C94BRL 9282942 IC50 = 1400 nM T84173 CR65TJ 9815399 IC50 = 29300 nM T84173 CMBS31 9859470 IC50 > 1000000 nM T84173 C0X2JQ 9881659 IC50 = 18500 nM T84173 C8CDL3 9882040 IC50 = 4000 nM T84173 C71BKL 9893924 IC50 = 360 nM T84173 C93DSQ 9989541 IC50 = 16700 nM T84173 CJ6TV8 10011928 IC50 = 500000 nM T84173 COC14Z 10039700 Ki = 83000 nM T84173 CZT1D2 10080697 Ki = 12800 nM T84173 C3O2JI 10093000 IC50 = 500 nM T84173 CE9XP3 10240946 IC50 = 54000 nM T84173 C98VYS 10313337 Ki = 199000 nM T84173 CL68SK 10319782 IC50 > 500000 nM T84173 CICJ52 10351835 Ki = 780000 nM T84173 C51PID 10352906 IC50 = 487000 nM T84173 C87EVT 10385642 IC50 > 500000 nM T84173 CB2NK4 10554498 IC50 = 2100 nM T84173 C4EIQ1 10559162 Ki = 98000 nM T84173 CX5QA1 10739903 IC50 > 500000 nM T84173 CA8C1Y 10752481 IC50 > 500000 nM T84173 CU1NP8 10788794 IC50 > 500000 nM T84173 C7GTH0 10820691 Ki = 110 nM T84173 CX9LI6 10844524 IC50 = 113000 nM T84173 C7R9UB 10932614 IC50 = 400000 nM T84173 C4KE9Z 11009466 IC50 = 100000 nM T84173 CWRD54 11062529 IC50 > 500000 nM T84173 CKH51F 11116404 Ki = 380000 nM T84173 CC4N0X 11258014 IC50 = 2000 nM T84173 CBF7L6 11744779 Ki = 42000000 nM T84173 CB9O8P 11773821 IC50 = 970000 nM T84173 CW28RN 12103488 Ki = 25 nM T84173 C12BNS 12766473 IC50 = 80000 nM T84173 C6M1GJ 12852767 Ki = 716000 nM T84173 CD18ZU 12910720 Ki = 500 nM T84173 CO9FE0 13880378 IC50 = 7780 nM T84173 CB7I6T 14752275 Ki = 1100 nM T84173 C1GEZ3 15999877 Ki = 120 nM T84173 CM9W3X 16002169 Ki = 184 nM T84173 CD0NR4 16003777 Ki = 121 nM T84173 CF1I7Z 16046245 IC50 = 11000 nM T84173 CQ03DX 16100284 IC50 = 507000 nM T84173 C20XPV 16100285 IC50 = 18000 nM T84173 C4SEC5 16100286 IC50 = 94000 nM T84173 CH90GF 16100287 IC50 = 393000 nM T84173 CQ0U4X 16355345 IC50 = 33210 nM T84173 C6EDP2 16759188 Ki = 55 nM T84173 C9IMC2 16759189 Ki = 514 nM T84173 CO2WR6 16759190 Ki = 122000 nM T84173 CIX5O8 17391397 IC50 = 720 nM T84173 C3S2UX 17518657 IC50 = 821 nM T84173 CHR32F 17546054 IC50 = 27 nM T84173 CQ04HS 17757274 IC50 = 330 nM T84173 COK9P5 21479008 IC50 = 4890 nM T84173 CM8SR5 21808535 IC50 = 405 nM T84173 CZ21NH 23622616 IC50 > 1000000 nM T84173 C54KMG 23647981 IC50 = 4200 nM T84173 CNB45K 23648009 IC50 = 7770 nM T84173 CQ5L3K 23648010 IC50 = 20700 nM T84173 CDUF21 23648011 IC50 = 6800 nM T84173 CAYB97 23648012 IC50 = 31100 nM T84173 CYK40M 23648013 IC50 = 6100 nM T84173 CJA9T5 23648014 IC50 = 18800 nM T84173 CW9EJ8 23648015 IC50 = 7750 nM T84173 CD94FU 23648016 IC50 = 2310 nM T84173 CG06QD 23648017 IC50 = 3940 nM T84173 CY8VL5 23648018 IC50 = 10040 nM T84173 C2Z6JH 23648019 IC50 = 28970 nM T84173 CN25MH 23648020 IC50 = 6690 nM T84173 CFOW76 23648021 IC50 = 1080 nM T84173 C3IP6A 23648022 IC50 = 8250 nM T84173 C63BFA 23648023 IC50 = 8800 nM T84173 CT9PR2 23648024 IC50 = 2000 nM T84173 C9DF0Y 23648025 IC50 = 770 nM T84173 C2NC6V 23648026 IC50 = 21670 nM T84173 CD3F8V 23648027 IC50 = 31400 nM T84173 CU9K5I 23648028 IC50 = 3340 nM T84173 CW4BH9 23648029 IC50 = 2390 nM T84173 CMHO50 23648030 IC50 = 1530 nM T84173 C6O5BZ 23648031 IC50 = 4900 nM T84173 CE7Z5U 23648032 IC50 = 2650 nM T84173 CAU8V5 23648033 IC50 = 2220 nM T84173 CCT73M 23648034 IC50 = 730 nM T84173 CF8EW3 23648035 IC50 = 370 nM T84173 CK8FT0 23648036 IC50 = 960 nM T84173 C6LA7B 23648037 IC50 = 3440 nM T84173 CH37FX 23648038 IC50 = 1040 nM T84173 CQ1V2E 25010186 IC50 = 700000 nM T84173 CL3Y5J 25010362 IC50 = 50000 nM T84173 CMKG19 31408646 IC50 = 4290 nM T84173 C57YWE 40225210 IC50 = 8900 nM T84173 CM7LJ5 44138544 IC50 = 46000 nM T84173 CJ2KC8 44138545 IC50 > 500000 nM T84173 CU70TS 44140356 IC50 = 295000 nM T84173 CAY6K5 44140485 IC50 > 500000 nM T84173 C80TMH 44267363 IC50 > 500000 nM T84173 CFM53I 44322630 IC50 > 300000 nM T84173 C9SB6W 44322665 IC50 = 200 nM T84173 C76PYN 44322883 IC50 = 211000 nM T84173 CF15IC 44322890 IC50 > 300000 nM T84173 CZAU45 44338547 Ki = 42000 nM T84173 C4R6EN 44338548 Ki = 900 nM T84173 CYBM80 44367875 IC50 > 1000000 nM T84173 CF7H4C 44368231 IC50 = 80000 nM T84173 C75BDZ 44368232 IC50 > 1000000 nM T84173 CS5ZN1 44368239 IC50 = 530000 nM T84173 CN5SX6 44377797 Ki = 800000 nM T84173 CLC70I 44377855 Ki = 8000000 nM T84173 C2XIE3 44377856 Ki = 20000000 nM T84173 C1Y6IA 44378051 Ki = 4000000 nM T84173 CLYZ61 44378065 Ki = 4500000 nM T84173 C4KHT0 44450759 Ki = 556 nM T84173 CCS5Z8 44450760 Ki = 23400 nM T84173 CKFL06 44565995 IC50 = 102000 nM T84173 CFHW02 44566012 IC50 = 175000 nM T84173 C26SVT 44566013 IC50 > 500000 nM T84173 C8GEN6 44566014 IC50 > 500000 nM T84173 COA0T6 44566015 IC50 > 500000 nM T84173 CP9C5R 44566016 IC50 = 127000 nM T84173 CYF3Q8 44566017 IC50 > 500000 nM T84173 C36HAV 44566018 IC50 = 253000 nM T84173 CB0Q6M 44566033 IC50 = 463000 nM T84173 C9O7DM 44566034 IC50 > 500000 nM T84173 C4E1IU 44566035 IC50 = 285000 nM T84173 CO19RL 44566036 IC50 > 500000 nM T84173 CX81GY 44566037 IC50 > 500000 nM T84173 CQ3SU2 44566055 IC50 > 500000 nM T84173 CA9V5Q 44566056 IC50 > 500000 nM T84173 CQ3SX9 44820249 IC50 = 200 nM T84173 CY74VL 44820542 IC50 = 45000 nM T84173 CB9RN5 44820543 IC50 = 2800 nM T84173 C4NG5O 44820544 IC50 = 46000 nM T84173 CF5I4L 44820545 IC50 = 1300 nM T84173 CB9X0Y 44820546 IC50 = 7300 nM T84173 C3XEY7 44820548 IC50 = 18300 nM T84173 CXL7R3 44820550 IC50 = 1200 nM T84173 CH3QT8 44820553 IC50 = 4000 nM T84173 C2S1XM 44820554 IC50 = 5800 nM T84173 CV6K5X 44820557 IC50 = 1300 nM T84173 CSO3P6 44820562 IC50 = 8200 nM T84173 CKRO61 44820563 IC50 = 18000 nM T84173 CE52UW 44820565 IC50 = 2000 nM T84173 CZT2A4 44820568 IC50 = 1000 nM T84173 CTSR92 44820569 IC50 = 2800 nM T84173 C4XI6P 44820570 IC50 = 800 nM T84173 CG5BL3 45102053 IC50 = 400 nM T84173 C2MO4N 45379774 Ki = 1 nM T84173 CDBC15 46867403 IC50 = 177827.94 nM T84173 CSG58C 46867528 IC50 = 223.87 nM T84173 CDI51T 46867529 Ki = 90 nM T84173 C06XNP 46867530 IC50 = 30 nM T84173 CZS29I 46867531 Ki = 80 nM T84173 CEY20W 46867532 Ki = 2400 nM T84173 CN5W6V 46867533 IC50 = 10715.19 nM T84173 CA18GU 46867661 IC50 = 1100 nM T84173 CQ5K9X 46867662 IC50 = 165958.69 nM T84173 CDNA73 46867663 IC50 = 11000 nM T84173 CD4JE2 46867664 IC50 = 4900 nM T84173 CQ19NU 46867665 IC50 = 257000 nM T84173 CE4KM7 46867666 IC50 = 18200 nM T84173 CNB14P 46867950 IC50 = 1200 nM T84173 CFY3Z7 46884603 IC50 = 147000 nM T84173 CX7E9P 46884604 IC50 = 43000 nM T84173 CDPL45 46889930 Ki = 300 nM T84173 CT23MN 51346766 IC50 = 12000 nM T84173 C6W5QS 52937504 Ki = 50 nM T84173 C60ZMG 52937505 IC50 = 237000 nM T84173 C9C7PW 52937506 IC50 = 66500 nM T84173 CWNY52 52937507 Ki = 770 nM T84173 CKW78O 52937508 IC50 = 10300 nM T84173 C0SK1N 52937608 IC50 = 12200 nM T84173 CBI17J 52937609 Ki = 1050 nM T84173 C8WQY5 52937610 Ki = 290 nM T84173 C7MZN8 52937611 IC50 = 35900 nM T84173 CAV3Z4 52937612 IC50 = 30900 nM T84173 C2QNA9 52937613 IC50 = 17300 nM T84173 C2GDN1 52937710 IC50 = 114000 nM T84173 CKY48T 52937711 IC50 = 10000 nM T84173 CQC41J 52937712 IC50 = 4320 nM T84173 C1U9HP 52937713 IC50 = 134000 nM T84173 CRHA98 52937714 Ki = 50 nM T84173 CX8NU3 52937715 IC50 = 466000 nM T84173 CQ0IY5 52937812 IC50 = 181000 nM T84173 C1LFC2 52937813 IC50 = 44500 nM T84173 C9N3MH 52937814 IC50 = 453000 nM T84173 CZ9XG6 52937815 IC50 = 325000 nM T84173 C65VST 52937816 IC50 = 5800 nM T84173 CZXI81 52937817 Ki = 890 nM T84173 C0SHU1 53317039 IC50 = 100000 nM T84173 C3YTE7 53317797 IC50 = 1750 nM T84173 CW28BO 53317798 IC50 = 40000 nM T84173 CWO7R2 53319114 IC50 = 500 nM T84173 C7VE6K 53319115 IC50 = 95000 nM T84173 C26RAJ 53320432 IC50 = 25000 nM T84173 CDAG25 53320433 IC50 > 1000000 nM T84173 C1ITM7 53321623 IC50 = 5400 nM T84173 CKHS34 53323067 IC50 = 705000 nM T84173 CYZX65 53323068 IC50 = 500 nM T84173 C2P5VF 53323483 IC50 > 1000000 nM T84173 CC46VH 53323661 IC50 = 60000 nM T84173 C1F7VA 53324417 IC50 = 100000 nM T84173 CGI17Z 53325719 IC50 = 30000 nM T84173 CZ4M6X 53325720 IC50 = 15000 nM T84173 C9VQ4F 53475226 Ki = 26 nM T84173 CQ04MF 56679802 Ki = 640000 nM T84173 CI9QC1 57341105 Ki = 450 nM T84173 CCX92D 57341107 Ki = 2700 nM T84173 COK1H5 57341110 Ki = 180 nM T84173 CAT3M0 57341112 Ki = 18 nM T84173 CQH9O2 57341114 Ki = 1.8 nM T84173 C3ECB7 57341116 Ki = 0.4 nM T84173 CQ1W6M 57341118 Ki = 76 nM T84173 CHT46N 57341120 Ki = 29 nM T84173 CQ8EC2 57341301 Ki = 4.4 nM T84173 CIP6O7 57341303 Ki = 6 nM T84173 CI39PZ 57341305 Ki = 4 nM T84173 CM59TH 57341307 Ki = 19 nM T84173 CQTP73 57341309 Ki = 3 nM T84173 CDH43T 57341311 Ki = 200 nM T84173 CZB17P 57341313 Ki = 12 nM T84173 CW6E1H 57341315 Ki = 30 nM T84173 C2SU4V 57341493 Ki = 250 nM T84173 C45FPH 57522037 IC50 = 780 nM T84173 CCF4G8 57522149 IC50 = 25 nM T84173 CJA14I 57522151 IC50 = 670 nM T84173 C6QIV0 57522153 IC50 = 170 nM T84173 CJ5U8K 57522155 IC50 = 19 nM T84173 CYEF31 57522157 Ki = 1 nM T84173 CI7FY4 57522159 IC50 = 120 nM T84173 C6ZYJ7 57522161 Ki = 820 nM T84173 CB4Z1A 57784577 IC50 = 60 nM T84173 CEM75P 60200911 IC50 = 11400 nM T84173 CCDK60 70681086 IC50 = 144000 nM T84173 CF9IE1 70683209 Ki = 700 nM T84173 CAD68M 70697642 IC50 = 19 nM T84173 C3VDS2 71299592 IC50 = 62000 nM T84173 CWPA60 71573724 IC50 > 1000000 nM T84173 C8VNE3 71717833 Ki = 5500000 nM T84173 CLJ89G 71770658 Ki = 1100 nM T84173 C4OQP2 71770659 Ki = 400 nM T84173 CBEP89 71770660 Ki = 1000 nM T84173 CG50PY 71770661 Ki = 400 nM T84173 CRX3F8 71770662 Ki = 3200 nM T84173 C7Z5PW 71770663 Ki = 71 nM T84173 C1YW3X 71770782 Ki = 4100 nM T84173 CID1P7 86298573 Ki = 34000 nM T84173 C9C3SK 86298574 Ki = 7.5 nM T84173 C6A9NO 90664973 IC50 = 81 nM T84173 C39TCQ 90665098 IC50 = 44400 nM T84173 C6ZP7C 90667059 Ki = 45000 nM T84173 CJ05EQ 90667060 Ki = 250 nM T84173 C2NXA4 101882899 IC50 = 300 nM T84173 C05DUA 101882900 IC50 = 6000 nM T84173 CU1NL5 118411065 IC50 = 200000 nM T84173 CH5U7F 118411068 IC50 = 100 nM T84173 C8X6RN 118411069 IC50 = 8000 nM T84173 C16QGB 118411070 IC50 = 20000 nM T84173 CD76NI 118411071 IC50 = 200 nM T84173 C9LGB3 118411072 IC50 = 250 nM T84173 CAR82K 118411073 IC50 = 400 nM T84173 CGXZ37 118411074 IC50 = 200 nM T84173 C8G3LO 118411076 IC50 = 1250 nM T84173 CB72ZY 118411077 IC50 = 125 nM T84173 C97IKP 118411079 IC50 = 3000 nM T84173 CV78UK 118411080 IC50 = 1500 nM T84173 CC84LW 118411081 IC50 = 2000 nM T84173 C2CF0W 118411108 IC50 = 5000 nM T84173 C89IWU 118411135 IC50 = 600 nM T84173 C5PIW8 118411136 IC50 = 600 nM T84173 CY83DV 118411140 IC50 = 250 nM T84173 CFH4O0 118411147 IC50 = 2500 nM T84173 CH7BA2 118411149 IC50 = 6000 nM T84173 CUYO63 118411153 IC50 = 15000 nM T84173 CZ7C5P 118718695 Ki = 2.4 nM T84173 C6GQ9L 118718696 Ki = 2.1 nM T84173 C80DCJ 118718742 Ki = 100 nM T84173 CLEP03 118718743 Ki = 150 nM T84173 C4O5TI 118718744 Ki = 100 nM T84173 C8H9CL 118718745 Ki = 1.2 nM T84173 CX1R5M 118718746 Ki = 550 nM T84173 C92EHU 118719203 Ki = 2100 nM T84173 C8PD0C 118719204 Ki = 66000 nM T84173 CMB63J 118719880 IC50 = 1500 nM T84173 CQ6CG3 118719881 IC50 = 500 nM T84173 C5N8JX 118719882 IC50 = 200 nM T84173 CL6Y0C 118719883 IC50 = 500 nM T84173 C53BCZ 118719884 IC50 = 400 nM T84173 C8G4SD 118719885 IC50 = 2500 nM T84173 CP0E3J 118719886 IC50 = 300 nM T84173 C8EXK9 118719887 IC50 = 1000 nM T84173 CHX93Q 118719888 IC50 = 10000 nM T84173 CN6TK0 118719889 IC50 = 500 nM T84173 CL97RN 118719890 IC50 = 60000 nM T84173 C60DKA 118719891 IC50 = 40000 nM T84173 C79GKI 118719892 IC50 = 12000 nM T84173 C5HZB0 118719893 IC50 = 5000 nM T84173 CJI04K 118719894 IC50 = 25000 nM T84173 C6OML9 118719895 IC50 = 15000 nM T84173 C1P9FV 118719896 IC50 = 10000 nM T84173 C86SLH 118719897 IC50 = 50000 nM T84173 CDTA82 118719898 IC50 = 10000 nM T84173 CXOU16 118719899 IC50 = 50000 nM T84173 C3FD9I 118719900 IC50 = 600000 nM T84173 CD56OM 118719901 IC50 = 15000 nM T84173 C3WIV2 118719902 IC50 = 250 nM T84173 CI1OS6 118719903 IC50 = 70 nM T84173 CSTV68 118719904 IC50 = 2500 nM T84173 CX4WV8 118719905 IC50 = 350 nM T84173 C1D3IO 118719906 IC50 = 700 nM T84173 CPVS50 118719907 IC50 = 400 nM T84173 CP9E1B 118719908 IC50 = 250 nM T84173 CHP35O 118719909 IC50 = 600 nM T84173 CZC89F 118719910 IC50 = 500 nM T84173 CE72DG 118719911 IC50 = 800 nM T84173 CCU4F2 118719912 IC50 = 800 nM T84173 CZ0PY7 118719913 IC50 = 500 nM T84173 C5JQ8G 118719914 IC50 = 250 nM T84173 C1MGA5 118719915 IC50 = 3000 nM T84173 CT6GP0 118719916 IC50 = 2000 nM T84173 C1SJU6 118719917 IC50 = 10000 nM T84173 CR67QX 118719918 IC50 = 3000 nM T84173 CC8N6I 118719919 IC50 = 300 nM T84173 C1WON3 118720302 IC50 = 400000 nM T84173 C0ZOT7 118720303 IC50 = 300 nM T84173 C81YUI 118720304 IC50 = 10000 nM T84173 CXI04D 118720305 IC50 = 10000 nM T84173 CG7JV9 118720306 IC50 = 20000 nM T84173 CR4S5Y 118720307 IC50 = 500000 nM T84173 CG9Q8E 118720308 IC50 = 12500 nM T84173 C8VC2U 118725788 IC50 = 33000 nM T84173 CO8JN9 118725789 IC50 = 230000 nM T84173 CX58QA 118725791 IC50 = 27000 nM T84173 C9I4RN 118725793 IC50 = 420000 nM T84173 CERW05 124168022 IC50 = 234 nM T84173 C02WIV 124168024 IC50 = 2140 nM T84173 C9BJ2O 124168025 IC50 = 8.3 nM T84173 C6P3RM 124168030 IC50 = 8.7 nM T84173 CW3EK7 124168033 IC50 = 4240 nM T84173 CG3WL1 124168088 IC50 = 430 nM T84173 CIG6O5 124168091 IC50 = 8.2 nM T84173 CK6HT0 124168092 IC50 = 2840 nM T84173 CZH9E8 124168098 IC50 = 8380 nM T84173 C8XE5C 124168100 IC50 = 926 nM T84173 C06QNJ 124168101 IC50 = 9.9 nM T84173 CV93ME 124168197 IC50 = 282 nM T84173 CA3Y1Q 124168198 IC50 = 5870 nM T84173 CNG3R2 124168199 IC50 = 891 nM T84173 CIH2U3 124168213 IC50 = 7300 nM T84173 C1AVE2 124168347 IC50 = 251 nM T84173 C7X6HL 124168348 IC50 = 5.2 nM T84173 C4M8XR 124168350 IC50 = 1880 nM T84173 C5XK9B 124168417 IC50 = 1530 nM T84173 CTH4O8 124168418 IC50 = 1280 nM T84173 CTC6Y5 124168420 IC50 = 9.4 nM T84173 C0F4DS 124168422 IC50 = 2540 nM T84173 CA82QT 124168429 IC50 = 9940 nM T84173 CCN6T5 124168443 IC50 = 126 nM T84173 CFP31U 124168444 IC50 = 857 nM T84173 C25FIC 124168445 IC50 = 872 nM T84173 C10UXO 124168446 IC50 = 431 nM T84173 CC74EP 127030046 Ki = 17370 nM T84173 CVA3Q4 127031609 IC50 = 5750 nM T84173 C89KHP 127031610 Ki = 1520 nM T84173 C7XRS6 127031611 IC50 = 21500 nM T84173 CSH65U 127031612 Ki = 140 nM T84173 CFS38P 127031892 Ki = 11550 nM T84173 CK0C8H 127031893 IC50 = 1430 nM T84173 CC80UH 127031894 Ki = 12340 nM T84173 C7XI4U 127032159 Ki = 8120 nM T84173 CY71AC 127032421 Ki = 640 nM T84173 C3U8GQ 127033032 Ki = 50 nM T84173 CD0IP7 127034618 IC50 > 1000000 nM T84173 C76JWP 127034620 IC50 > 1000000 nM T84173 CAF9D8 127034622 IC50 > 1000000 nM T84173 C1GX2A 127034624 IC50 > 1000000 nM T84173 CG0M8L 127034626 IC50 > 1000000 nM T84173 C1KA0S 127034628 IC50 > 1000000 nM T84173 CWDC64 127034630 IC50 > 1000000 nM T84173 CV03JM 127034632 IC50 > 1000000 nM T84173 CHY10W 127035143 IC50 > 1000000 nM T84173 CO3R1K 127035145 IC50 > 1000000 nM T84173 CLSC85 127035326 IC50 > 1000000 nM T84173 CO52UV 127035677 IC50 > 1000000 nM T84173 C5S0JI 127036664 IC50 > 1000000 nM T84173 CW2DX5 127037636 IC50 > 1000000 nM T84173 C0N7KM 134131863 IC50 = 6800 nM T84173 C5BW3X 134134697 IC50 = 122 nM T84173 CRIE82 134137830 IC50 = 121000 nM T84173 CPA9Z7 134138587 IC50 > 1000000 nM T84173 C15KGS 134143870 IC50 = 21.1 nM T84173 CKU2P9 134144115 IC50 = 788000 nM T84173 CG6ES5 134146186 IC50 = 35 nM T84173 CYNV84 134148190 IC50 = 8600 nM T84173 CWH70S 134149179 IC50 = 12400 nM T84173 CJ4V8N 134150037 IC50 = 29.4 nM T84173 CIWE29 134152584 IC50 = 12.5 nM T84173 C7Y2ZL 134152833 IC50 = 4100 nM T84173 CP2GU6 134154157 IC50 = 4900 nM T84173 C2XRJ7 134154906 IC50 = 168 nM T84173 CSQT91 134157313 IC50 = 7300 nM T84173 C3P9GJ 137634997 Ki = 10300 nM T84173 CQT81G 137640259 Ki = 19 nM T84173 C2FY5W 137644530 Ki = 54200 nM T84173 C40OGM 137645711 Ki = 1 nM T84173 CRX18K 137647938 Ki = 10700 nM T84173 C43TEW 137649273 Ki = 900 nM T84173 CIE71B 137651681 Ki = 300 nM T84173 CIT85R 137654457 Ki = 600 nM T84173 C0ZT7D 137659840 Ki = 90 nM T84173 CYKH62 137661141 Ki = 123000 nM T84173 CT0Q8H 145965670 IC50 = 187000 nM T84173 CK4QZ0 145967390 IC50 = 11000 nM T84173 CXZH98 145971016 IC50 = 31000 nM T84173 C58SHF 145972263 IC50 = 19000 nM T84173 CD5G9J 145977376 IC50 = 19000 nM T84173 CE40SO 145978797 IC50 = 28000 nM T84173 C1MD8E 145981653 IC50 = 25 nM T84173 CP2VA7 145991605 IC50 = 2561 nM T84173 C4YB1L 155511412 IC50 = 603000 nM T84173 C7JG9T 155527701 IC50 = 136000 nM T84173 D00MFZ 44578588 IC50 = 9000 nM T84173 D01HDD 983732 IC50 > 500000 nM T84173 D01TOR 667555 IC50 = 5770 nM T84173 D04QWD 7027 Ki = 30000 nM T84173 D05CEM 5311371 IC50 = 600 nM T84173 D06YQR 46884602 IC50 = 560 nM T84173 D09IWI 46229705 IC50 = 1650 nM T84173 D0B1WB 11988371 Ki = 2.2 nM T84173 D0N9IX 9822159 IC50 = 100 nM T84173 D0Q7SF 46229704 IC50 = 350 nM T84173 D0R2BA 445248 Ki = 4280 nM T84173 D0R4JZ 46866608 IC50 = 19 nM T84173 D0R8TR 445612 Ki = 1300 nM T84173 D0S4DV 124434 IC50 = 1000 nM T84173 D0SQ1T 10261406 Ki = 200 nM T84173 D0X6LK 10823890 IC50 > 500000 nM T94119 D09XZB 123631 IC50 > 50000 nM T94119 D0B3HD 2519 IC50 = 75000 nM T94119 D0E6XR 3062316 IC50 = 30000 nM T94119 D0F8RA 2153 IC50 = 75000 nM T94119 D0J5VR 11625818 IC50 = 1.2 nM T94119 D0R0MW 5329102 IC50 = 12000 nM T94119 D0RU0O 50905713 IC50 < 0.5 nM T94119 D0S5LD 135565596 IC50 < 0.7 nM T94119 D0W5HK 216239 IC50 > 50000 nM T94119 D00UZR 5330286 IC50 > 10000 nM T94119 D01PGR 16123056 IC50 = 43 nM T94119 D01QSO 16654980 IC50 = 110 nM T94119 D03BHZ 52913813 IC50 = 12 nM T94119 D03EZE 25167777 IC50 = 2.5 nM T94119 D03FOP 68947304 IC50 = 10.9 nM T94119 D03IJO 11618268 IC50 = 12.7 nM T94119 D03KAC 1893730 IC50 = 36 nM T94119 D03LWG 53235510 IC50 > 9000 nM T94119 D03XAQ 49784945 IC50 = 500 nM T94119 D06GUA 49784002 Ki = 0.1259 nM T94119 D07EHV 44814409 IC50 > 9100 nM T94119 D07HPJ 11476171 IC50 > 9100 nM T94119 D08QGT 17755052 IC50 = 3 nM T94119 D0C3ZR 10427712 IC50 = 235 nM T94119 D0D8JB 44516953 IC50 = 6 nM T94119 D0I3LO 91933883 IC50 = 23 nM T94119 D0LG7X 86291103 IC50 = 24.5 nM T94119 D0O1LD 11647372 IC50 = 3 nM T94119 D0O6VZ 25254071 IC50 = 6.7 nM T94119 D0O8SJ 72950888 IC50 = 6.2 nM T94119 D0TU7B 58507717 IC50 = 451 nM T94119 D0U3DP 46912230 IC50 = 37 nM T94119 D0UP1Z 51001932 Ki = 0.12 nM T94119 D0VG0D 11977753 IC50 = 5 nM T94119 D0W7HE 56649450 IC50 = 290 nM T94119 D0XD4I 118502708 IC50 = 270 nM T94119 D0Y2NS 70798655 IC50 = 13900 nM T94119 D03BNU 59604787 IC50 > 5000 nM T94119 D0C9JZ 58111426 IC50 = 3.4 nM T94119 D0E0YY 53235521 IC50 < 50 nM T94119 D05HIJ 135565159 IC50 = 468 nM T94119 D09SFV 3973 IC50 = 500 nM T94119 D0D0QA 44137675 IC50 = 80 nM T94119 D0P1JI 312145 IC50 = 4 nM T94119 C3FRX9 131989 IC50 = 65700 nM T94119 C05RDN 566479 IC50 = 6800 nM T94119 CY3D4G 617191 IC50 = 3887 nM T94119 CS5O7B 622000 IC50 > 40000 nM T94119 CXC3V1 622262 IC50 = 701 nM T94119 CU73NO 736009 IC50 > 83300 nM T94119 C0L5VC 946390 IC50 = 900 nM T94119 CWOQ49 1627922 IC50 = 90 nM T94119 CKCW93 2612441 IC50 > 100000 nM T94119 C09VKD 2816900 IC50 = 36800 nM T94119 CK79GO 2988969 IC50 > 100000 nM T94119 C1O4KS 4416330 IC50 > 25000 nM T94119 CIN5F7 4904109 IC50 <= 10000 nM T94119 C1YJM9 4912089 IC50 > 83300 nM T94119 CE74CV 5059890 IC50 = 100000 nM T94119 C2OZ0W 6484194 IC50 = 18000 nM T94119 CK2IR4 6852165 IC50 = 180 nM T94119 CE1Y8A 9815659 IC50 = 5100 nM T94119 CJ79RC 9879653 IC50 = 3 nM T94119 CC4F8I 10021687 IC50 = 800 nM T94119 CZM84H 10066542 IC50 = 800 nM T94119 C2W9ED 10269329 IC50 = 230 nM T94119 C7SFI1 10296883 IC50 > 10000 nM T94119 C32NQS 10357196 IC50 = 4204 nM T94119 CAZT53 10475366 IC50 = 29 nM T94119 CL8YE3 11230964 IC50 = 2900 nM T94119 C8Y6IM 11234514 IC50 = 98 nM T94119 CK65NF 11418892 Ki = 2900 nM T94119 CL3Z4O 11419728 IC50 = 16 nM T94119 CYBD21 11428504 IC50 = 140 nM T94119 CI2YV6 11474717 IC50 = 197 nM T94119 CHJ30L 11492951 IC50 > 20000 nM T94119 CR41FO 11502414 IC50 = 6 nM T94119 C0O4SQ 11522078 IC50 > 5000 nM T94119 C7HMO6 11526786 IC50 = 11 nM T94119 C38YWS 11541283 IC50 = 1 nM T94119 C1VA4C 11543481 IC50 = 810 nM T94119 CN2MS6 11562853 IC50 = 25.12 nM T94119 CMVQ43 11576772 IC50 = 0.9 nM T94119 C8K6VJ 11584055 Ki = 1.1 nM T94119 CEHZ82 11599141 IC50 = 39.81 nM T94119 C1ZPM5 11630874 IC50 = 20000 nM T94119 CYU3J9 11634899 IC50 = 1.7 nM T94119 CP04JC 11666231 IC50 = 16.1 nM T94119 C48YXV 11677284 Ki = 4.9 nM T94119 CY8C9P 11751126 IC50 = 201 nM T94119 CBR6D5 11955693 IC50 = 187 nM T94119 C60DBM 11998444 IC50 = 31710 nM T94119 C5FTB0 11998445 IC50 = 1176 nM T94119 C68WMR 11998447 IC50 = 26240 nM T94119 CYL24B 11998448 IC50 = 5973 nM T94119 CNPI54 11998563 IC50 = 2525 nM T94119 C6AK0Y 11998564 IC50 = 1392 nM T94119 CMVA72 11998565 IC50 = 126 nM T94119 CJ3YP8 11998685 IC50 = 2124 nM T94119 CV8PB5 11998690 IC50 = 614 nM T94119 CB9T1H 11998803 IC50 = 35 nM T94119 C59SKD 11999032 IC50 = 18 nM T94119 CY7A0T 14638904 IC50 = 12500 nM T94119 CH1DJ6 16036739 IC50 = 16 nM T94119 CVN8B2 16049456 IC50 = 251.19 nM T94119 CW2XK6 16050925 IC50 = 530 nM T94119 CW5FD8 16081736 IC50 = 1482 nM T94119 CV9US5 16736978 IC50 = 5300 nM T94119 CF6JS9 16757570 IC50 = 340 nM T94119 CB19TH 16757576 IC50 = 1000 nM T94119 C1NZC7 16757579 IC50 = 166 nM T94119 C1SN9M 17756679 IC50 >= 100000 nM T94119 CVDL81 22036885 IC50 = 0.65 nM T94119 C61ZGT 22135435 IC50 = 79432.82 nM T94119 CP05ZB 22346757 IC50 = 23000 nM T94119 C1F2TM 23582995 IC50 = 950 nM T94119 CEYL29 23585510 Ki = 740 nM T94119 COW91A 23586721 IC50 = 710 nM T94119 CBL37C 23642173 Ki = 4 nM T94119 C8J1SI 23642272 IC50 = 722 nM T94119 C29SFI 24768579 IC50 = 249 nM T94119 C72BSE 24804168 IC50 = 19952.62 nM T94119 C6Y5GV 24805152 IC50 = 19952.62 nM T94119 CL4C8H 24809743 IC50 = 3600 nM T94119 CP4G9Z 24855584 Ki = 3 nM T94119 CJV7D9 24855887 IC50 = 54 nM T94119 CM9C0R 24866805 IC50 = 6700 nM T94119 CB79YC 24905143 IC50 = 250 nM T94119 C2DC9J 24905144 IC50 = 800 nM T94119 CN6V8Z 24905145 IC50 = 27 nM T94119 CSB7P5 24905148 IC50 = 2300 nM T94119 CGSF21 24905149 IC50 = 3 nM T94119 CVDG02 24905150 IC50 = 10200 nM T94119 CWH6C5 24905152 IC50 = 6 nM T94119 C0HE2Q 24905153 IC50 = 4 nM T94119 C7QSC9 24905154 IC50 = 680 nM T94119 CO9D0K 24905155 IC50 = 410 nM T94119 C5W9UR 24905157 IC50 = 140 nM T94119 CC1DA3 24905158 IC50 = 690 nM T94119 COW79F 24905159 IC50 = 650 nM T94119 CFPA53 24905160 IC50 = 640 nM T94119 C2O0JX 24905161 IC50 = 1400 nM T94119 CA72BE 24905162 IC50 = 210 nM T94119 CQN6X9 24905163 IC50 = 1900 nM T94119 CD4O1F 24905165 IC50 = 3700 nM T94119 CKL48T 24905166 IC50 = 1200 nM T94119 C76VYL 24905167 IC50 = 900 nM T94119 C7K5PU 24905168 IC50 = 125 nM T94119 CZ57ID 24905169 IC50 = 730 nM T94119 C2DHX9 24905170 IC50 = 1900 nM T94119 CSB96E 24905171 IC50 = 100000 nM T94119 CWZ0R2 24905172 IC50 = 1300 nM T94119 CY3B6M 24905175 IC50 = 281 nM T94119 CW1V0H 24905177 IC50 = 1900 nM T94119 CO6Y0L 24905178 IC50 = 37000 nM T94119 C60NQW 24905179 IC50 = 686 nM T94119 C4MO8B 24905180 IC50 = 677 nM T94119 COJI47 24905181 IC50 = 249 nM T94119 CS0B2C 24905182 IC50 = 72 nM T94119 C1H4BT 24905183 IC50 = 144 nM T94119 C4WHK9 24905184 IC50 = 2970 nM T94119 C7Q4MZ 24905185 IC50 = 2480 nM T94119 CS4IP1 24905186 IC50 = 130 nM T94119 C69QWO 24905187 IC50 = 1030 nM T94119 C85ANB 24905188 IC50 = 173 nM T94119 CNHD75 24905189 IC50 = 57 nM T94119 C9JUO2 24905190 IC50 = 2020 nM T94119 CPR03K 24905191 IC50 = 446 nM T94119 CTAG19 24905193 IC50 = 228 nM T94119 C7VJM5 24905194 IC50 = 643 nM T94119 CEP1L3 24905195 IC50 = 436 nM T94119 CP68ZD 24905196 IC50 = 429 nM T94119 C8Z0RJ 24905197 IC50 = 255 nM T94119 CN9RT0 24905198 IC50 = 1200 nM T94119 CHI78P 24905200 IC50 = 400 nM T94119 CO6PE8 24905201 IC50 = 340 nM T94119 CZ63HS 24905202 IC50 = 77 nM T94119 C2X0FC 24905203 IC50 = 120 nM T94119 C0WCE3 24905204 IC50 = 90 nM T94119 CNK50B 24905205 IC50 = 89 nM T94119 C12DPB 24905206 IC50 = 190 nM T94119 C8N0RH 24905207 IC50 = 3700 nM T94119 CYA5G2 24905208 IC50 = 56 nM T94119 CDV2B4 24905209 IC50 = 660 nM T94119 CEFK68 24905210 IC50 = 140 nM T94119 CUFP12 24905211 IC50 = 453 nM T94119 C0JG8L 24905212 IC50 = 966 nM T94119 CP47MK 24905213 IC50 = 18000 nM T94119 CB61QC 24905214 IC50 = 2300 nM T94119 CQ13ZI 24905215 IC50 = 3400 nM T94119 C6VI8F 24905216 IC50 = 123 nM T94119 CXNH25 24905217 IC50 = 85 nM T94119 C2PN9S 24905218 IC50 = 49 nM T94119 C9O2AL 24905219 IC50 = 110 nM T94119 CIT7U8 24905220 IC50 = 1800 nM T94119 CMD26S 24905221 IC50 = 37 nM T94119 C4R8WC 24905222 IC50 = 443 nM T94119 C47SHA 24905223 IC50 = 100 nM T94119 C1DY2R 24905224 IC50 = 142 nM T94119 CS0XF9 24905225 IC50 = 409 nM T94119 CG5VX2 24905226 IC50 = 100000 nM T94119 C57QEO 24905227 IC50 = 100000 nM T94119 C7CG5E 24905228 IC50 = 1000 nM T94119 CHP5D1 24905229 IC50 = 1700 nM T94119 CXP09S 24905230 IC50 = 120 nM T94119 CY7XG1 24905231 IC50 = 1500 nM T94119 C7JFQ2 24905232 IC50 = 375 nM T94119 C2JM1P 24905233 IC50 = 5200 nM T94119 CC3BF0 24905234 IC50 = 3900 nM T94119 CE57FI 24905235 IC50 = 3900 nM T94119 CUP20O 24905236 IC50 = 6300 nM T94119 CLC6Q2 24905237 IC50 = 1400 nM T94119 C9M1GI 24905238 IC50 = 213 nM T94119 CVD72F 24905239 IC50 = 68 nM T94119 CK38IZ 24905240 IC50 = 88 nM T94119 CO2V5E 24905241 IC50 = 2000 nM T94119 CZBA19 24905244 IC50 = 162 nM T94119 CQ8OI1 24905246 IC50 = 72000 nM T94119 C5URC6 24905247 IC50 = 1800 nM T94119 CZ2E9K 24905249 IC50 = 3000 nM T94119 C03SVO 24905250 IC50 = 9600 nM T94119 CIF2J5 24905251 IC50 = 280 nM T94119 CPTE58 24905252 IC50 = 1260 nM T94119 CX1JB8 24905253 IC50 = 5700 nM T94119 COZ3H7 24905254 IC50 = 29000 nM T94119 CDT1H9 24905255 IC50 = 11000 nM T94119 C54QKA 24905256 IC50 = 3100 nM T94119 CRU3P2 24905257 IC50 = 100000 nM T94119 C9U0JA 24905259 IC50 = 11000 nM T94119 CO4YS7 24905260 IC50 = 82000 nM T94119 CEG0B5 24905261 IC50 = 100000 nM T94119 C9VE5F 24905262 IC50 = 100000 nM T94119 C3I4HK 24905264 IC50 = 6300 nM T94119 C0VMI6 24905265 IC50 = 100000 nM T94119 CWE3V0 24905267 IC50 = 100000 nM T94119 CH4T3A 24905268 IC50 = 100000 nM T94119 CVT17Q 24905270 IC50 = 750 nM T94119 C6QDN7 24905271 IC50 = 2900 nM T94119 C6XHJ7 24905272 IC50 = 1200 nM T94119 CTB9A3 24905273 IC50 = 28000 nM T94119 C0NB1Q 24905274 IC50 = 21000 nM T94119 C9KQ0L 24905275 IC50 = 3000 nM T94119 C9O8QZ 24905277 IC50 = 7400 nM T94119 CP50RD 24905280 IC50 = 65 nM T94119 CG13ZM 24905281 IC50 = 252 nM T94119 CF0S6X 24905282 IC50 = 42 nM T94119 C5HBL0 24905284 IC50 = 3190 nM T94119 C2Z5DN 24905285 IC50 = 660 nM T94119 CL6GH8 24905286 IC50 = 198 nM T94119 CKYO98 24905287 IC50 = 220 nM T94119 CRNQ65 24905288 IC50 = 74 nM T94119 COD7I5 24905289 IC50 = 470 nM T94119 C4LP7E 24905290 IC50 = 210 nM T94119 CE9JC2 24905291 IC50 = 76 nM T94119 C2GI1R 24905292 IC50 = 473 nM T94119 CHW8C4 24905293 IC50 = 47 nM T94119 CQF0H1 24905294 IC50 = 10 nM T94119 CNO7X0 24905295 IC50 = 12 nM T94119 C5WRG7 24905296 IC50 = 17 nM T94119 CQ1S0U 24905297 IC50 = 276 nM T94119 C4UES7 24905298 IC50 = 177 nM T94119 CMS69P 24905299 IC50 = 6050 nM T94119 CC0U5M 24905300 IC50 = 103 nM T94119 CW7X6S 24905301 IC50 = 1985 nM T94119 C97IQV 24905302 IC50 = 142 nM T94119 CSJ47V 24905303 IC50 = 199 nM T94119 CPN74C 24905304 IC50 = 5470 nM T94119 C5CS3N 24905305 IC50 = 207 nM T94119 CK4XE9 24905307 IC50 = 172 nM T94119 CTU6Z3 24905308 IC50 = 1070 nM T94119 C9SQX1 24905309 IC50 = 193 nM T94119 CM75JP 24905310 IC50 = 514 nM T94119 C9Q2BJ 24905311 IC50 = 680 nM T94119 C9VUA1 24905312 IC50 = 203 nM T94119 CU3RS1 24905313 IC50 = 215 nM T94119 CYG3H2 24905314 IC50 = 213 nM T94119 CV5Q7O 24905315 IC50 = 58 nM T94119 C8SA3O 24905316 IC50 = 13 nM T94119 CI5MN3 24905317 IC50 = 20 nM T94119 CJ1P7K 24905318 IC50 = 12 nM T94119 C1T6YQ 24905319 IC50 = 15 nM T94119 CAU86X 24905320 IC50 = 49 nM T94119 C54ISY 24905321 IC50 = 3030 nM T94119 C2GE5I 24905322 IC50 = 1620 nM T94119 C8D6YK 24905323 IC50 = 4350 nM T94119 C5NZH9 24905324 IC50 = 1000 nM T94119 C9D6JR 24905325 IC50 = 777 nM T94119 CLZT41 24905326 IC50 = 150 nM T94119 CW8FD3 24905327 IC50 = 74 nM T94119 CHB7A2 24905328 IC50 = 1370 nM T94119 CA8EI3 24905329 IC50 = 716 nM T94119 CCQ0O7 24905330 IC50 = 197 nM T94119 CJ81AS 24905331 IC50 = 23 nM T94119 C8PW4H 24905332 IC50 = 41 nM T94119 C2Y5TF 24905333 IC50 = 112 nM T94119 CH9FL5 24905334 IC50 = 67 nM T94119 C1S0PC 24905335 IC50 = 120 nM T94119 C8N9MV 24905336 IC50 = 206 nM T94119 C9E8BJ 24905338 IC50 = 240 nM T94119 CX85AC 24905341 IC50 = 6900 nM T94119 CKZ80E 24905342 IC50 = 46 nM T94119 CO8SH1 24905343 IC50 = 48 nM T94119 C7IZL6 24905344 IC50 = 670 nM T94119 C43VSW 24936353 IC50 = 10 nM T94119 C83EUF 24937010 IC50 = 3 nM T94119 C72LWC 24937637 IC50 = 3.2 nM T94119 C6E3AN 24944519 IC50 = 0.5 nM T94119 CHI9W6 24944522 IC50 = 105.9 nM T94119 C98MEW 24946175 IC50 = 11 nM T94119 CC7H3U 24946706 IC50 = 0.7 nM T94119 C78NJE 24955795 IC50 = 549 nM T94119 C8P6NT 24956158 IC50 = 80 nM T94119 CJI29P 24956159 IC50 = 5731 nM T94119 CXV6R0 24968746 Ki = 7 nM T94119 C6C4RH 24993871 IC50 = 12 nM T94119 CEW91Q 25032963 IC50 = 4 nM T94119 CY50OT 25052783 IC50 = 32 nM T94119 CHR51O 25057242 IC50 = 61 nM T94119 CF8G3J 25095512 IC50 = 2 nM T94119 CD69RK 25097993 IC50 < 0.5 nM T94119 CLP07J 25110819 IC50 > 10000 nM T94119 CVM89J 25128663 IC50 = 5011.87 nM T94119 C4HRL9 25128667 IC50 = 1995.26 nM T94119 C4SWT5 25128668 IC50 > 79432.82 nM T94119 CIO6A4 25129024 IC50 > 100000 nM T94119 CLS7P0 25129381 IC50 = 6309.57 nM T94119 C9R2EA 25129383 IC50 = 31622.78 nM T94119 C4YZL9 25129386 IC50 = 5011.87 nM T94119 CDO9Q0 25129729 IC50 > 100000 nM T94119 CX86YV 25129734 IC50 > 19952.62 nM T94119 CA2K4U 25130429 IC50 = 501.19 nM T94119 C1J8KH 25132804 IC50 = 3162.28 nM T94119 CI04XW 25132806 IC50 = 31622.78 nM T94119 C5WC4L 25133141 IC50 > 31622.78 nM T94119 CSH37X 25133142 IC50 > 10000 nM T94119 CW3HN6 25133144 IC50 > 100000 nM T94119 C4LHV1 25165368 IC50 > 10000 nM T94119 C2CXH3 25165371 IC50 > 10000 nM T94119 CQWL59 25165372 IC50 > 10000 nM T94119 CL87JW 25165773 IC50 > 30000 nM T94119 CB89TL 25165774 IC50 > 10000 nM T94119 CFZI92 25165961 IC50 > 10000 nM T94119 CK2YI4 25168990 IC50 = 9332.54 nM T94119 C7G1ZM 25169579 IC50 = 250 nM T94119 CL81FJ 25169580 IC50 = 320 nM T94119 C8WL0Z 25169784 IC50 > 1000 nM T94119 CLR8M2 25169786 IC50 = 690 nM T94119 CL3UK2 25170000 IC50 > 1000 nM T94119 C6WCR7 25170003 IC50 = 120 nM T94119 C2RT9W 25170004 IC50 = 230 nM T94119 CSK97U 25170005 IC50 > 1000 nM T94119 C7AH2I 25170203 IC50 = 280 nM T94119 C2TEW6 25170204 IC50 > 1000 nM T94119 C5PTZ0 25170410 IC50 = 89 nM T94119 CLJR80 25171641 IC50 = 3400 nM T94119 C7ZQC2 25171642 IC50 = 700 nM T94119 C7AHP4 25171644 IC50 > 1000 nM T94119 CX6BL8 25171852 IC50 > 1000 nM T94119 C7TL2N 25171853 IC50 > 1000 nM T94119 C6BR3F 25171855 IC50 = 90 nM T94119 CMI85O 25171856 IC50 = 150 nM T94119 CUN9F3 25171857 IC50 = 170 nM T94119 CKY81J 25172061 IC50 > 1000 nM T94119 CC1D8V 25172062 IC50 = 49 nM T94119 C1L6GX 25172063 IC50 = 410 nM T94119 CFO08N 25172065 IC50 = 35 nM T94119 C8ZF0A 25172066 IC50 = 2000 nM T94119 CCW80B 25172270 IC50 > 1000 nM T94119 C9HUB6 25172271 IC50 = 310 nM T94119 CC60ZY 25172272 IC50 = 180 nM T94119 C54EGX 25172274 IC50 = 400 nM T94119 C5QVC7 25172275 IC50 = 200 nM T94119 CPW2D9 25172477 IC50 = 54 nM T94119 CVDC60 25172479 IC50 = 580 nM T94119 CI6W9H 25172661 IC50 = 9.3 nM T94119 CL5IC0 25172662 IC50 = 110 nM T94119 CDAO95 25172663 IC50 = 180 nM T94119 C8JC3P 25172664 IC50 = 8.6 nM T94119 CK38ER 25172665 IC50 = 16 nM T94119 C3JI1Y 25172666 IC50 = 37 nM T94119 CLW96O 25207689 IC50 = 6 nM T94119 CWP29U 25242324 IC50 = 16 nM T94119 C96OGS 25260915 IC50 = 64 nM T94119 CUR93V 25261554 IC50 > 10000 nM T94119 C3IDN0 25266674 IC50 = 1000 nM T94119 C2IM0O 39733146 IC50 = 7943.28 nM T94119 C1O8ZY 42596976 IC50 = 665 nM T94119 CO4PL8 42606076 IC50 > 100000 nM T94119 C20VGT 42606077 IC50 = 39000 nM T94119 C7N5EC 42606078 IC50 > 100000 nM T94119 CIF63E 42623219 IC50 = 6309.57 nM T94119 C3DNM9 42623223 IC50 = 1584.89 nM T94119 COR5I0 42623224 IC50 = 7943.28 nM T94119 CX1DC2 42623385 IC50 = 398.11 nM T94119 CR6N3I 42623632 IC50 > 6309.57 nM T94119 C4EM0W 42623869 IC50 = 1584.89 nM T94119 C5TY9Q 42623950 IC50 = 3162.28 nM T94119 C10RBA 42636535 IC50 = 1500 nM T94119 CKH08W 44123663 IC50 < 100 nM T94119 C3ROX1 44124863 Ki = 0.8 nM T94119 CI3K7H 44129042 IC50 = 4000 nM T94119 CIE0J3 44129043 IC50 = 7900 nM T94119 CUW85V 44129044 IC50 > 10000 nM T94119 C2B9DE 44129118 IC50 = 3800 nM T94119 C0R1PH 44129198 IC50 = 8100 nM T94119 C6LGD5 44129200 IC50 = 630 nM T94119 C03RLS 44129270 IC50 > 10000 nM T94119 CU4H1I 44129274 IC50 = 7400 nM T94119 C79QOC 44129275 IC50 = 1600 nM T94119 C0W3ZF 44129348 IC50 = 9200 nM T94119 CH6RO4 44129351 IC50 = 3300 nM T94119 CPAU59 44129353 IC50 = 1800 nM T94119 CN5O4I 44129429 IC50 = 810 nM T94119 C3ZSV2 44129432 IC50 = 1500 nM T94119 CM5U2I 44137407 IC50 = 190 nM T94119 CF17OS 44180029 IC50 = 4200 nM T94119 CHK8Z6 44180034 IC50 = 27 nM T94119 CEJ5F7 44180035 IC50 > 20000 nM T94119 CQNT23 44180155 IC50 > 50000 nM T94119 CIKM57 44180156 IC50 = 960 nM T94119 CBP2T3 44180157 IC50 = 7894 nM T94119 C9CGB4 44180282 IC50 > 50000 nM T94119 C2S5LC 44180395 IC50 = 26 nM T94119 C40NOQ 44180397 IC50 = 18 nM T94119 CTB46H 44180398 IC50 = 12 nM T94119 CE30IL 44180626 IC50 = 20 nM T94119 CRS2G3 44180853 IC50 = 14940 nM T94119 C2VZX7 44181492 IC50 = 2420 nM T94119 C7SYM2 44181493 IC50 > 50000 nM T94119 CB8KF1 44181494 IC50 > 23000 nM T94119 C5AI8R 44181598 IC50 > 30000 nM T94119 CK03RW 44181599 IC50 > 50000 nM T94119 CXL61J 44181600 IC50 = 784 nM T94119 C6TZK5 44181601 IC50 = 481 nM T94119 CCIV74 44181602 IC50 = 555 nM T94119 C36WUP 44181603 IC50 > 50000 nM T94119 CS2U7R 44181604 IC50 = 9807 nM T94119 CL6W0C 44181605 IC50 = 8936 nM T94119 CFD41Z 44181718 IC50 = 13830 nM T94119 C2RB1P 44181719 IC50 > 23000 nM T94119 CMC75I 44181720 IC50 = 1142 nM T94119 CWTS93 44181721 IC50 = 3998 nM T94119 CT1JL2 44181722 IC50 = 3732 nM T94119 CE9HO1 44181723 IC50 = 278 nM T94119 CFSB29 44181724 IC50 = 649 nM T94119 C13DKP 44219291 IC50 = 12 nM T94119 CMNC52 44225402 IC50 < 50 nM T94119 C6RDB9 44237450 IC50 > 100 nM T94119 C98MAL 44436951 IC50 = 5400 nM T94119 CD0ME6 44436952 IC50 > 10000 nM T94119 CR6ZU9 44436953 IC50 > 10000 nM T94119 CYK0T1 44436954 IC50 > 10000 nM T94119 CYV15O 44436955 IC50 > 10000 nM T94119 C3M4RN 44436961 IC50 > 10000 nM T94119 CA4SV2 44436964 IC50 > 10000 nM T94119 CO5FK1 44436967 IC50 > 10000 nM T94119 CRKU98 44436970 IC50 > 10000 nM T94119 C9V1SZ 44436971 IC50 > 10000 nM T94119 CZ4V2L 44436972 IC50 > 10000 nM T94119 COG34Q 44436976 IC50 > 10000 nM T94119 C4RAK8 44436979 IC50 = 9000 nM T94119 CXN93Q 44436980 IC50 > 10000 nM T94119 CX57RI 44436981 IC50 > 10000 nM T94119 C9ZML1 44454396 IC50 = 35 nM T94119 C4PR1L 44466962 Ki = 10 nM T94119 C30NZA 44475985 IC50 = 21 nM T94119 CAT8F7 44475986 IC50 = 1 nM T94119 CSR73H 44475987 IC50 = 7 nM T94119 CDAX92 44475988 IC50 = 40 nM T94119 CBH0S5 44475989 IC50 = 34 nM T94119 CW5A7L 44475990 IC50 = 0.5 nM T94119 CG9A5L 44511405 IC50 <= 10000 nM T94119 CFC65B 44539960 IC50 <= 10000 nM T94119 C03IGD 44540030 IC50 = 1584.89 nM T94119 C5LWU1 44540126 IC50 = 3981.07 nM T94119 CYD4Z8 44540130 IC50 = 1.995 nM T94119 CAT2R7 44540316 IC50 = 3162.28 nM T94119 C36NRP 44540403 IC50 <= 10000 nM T94119 C2T9GC 44540407 IC50 = 100 nM T94119 CQ4PE7 44540492 IC50 = 1000 nM T94119 CZ9GL8 44541044 IC50 = 12.59 nM T94119 C6L4SV 44545041 Ki = 4 nM T94119 CPCJ61 44554231 IC50 < 100 nM T94119 C0N2VK 44554233 IC50 < 100 nM T94119 C3VRO9 44557921 IC50 = 707.95 nM T94119 CN2O9S 44577591 IC50 > 20000 nM T94119 CRE61W 44577592 IC50 = 74 nM T94119 CH63GM 44577593 IC50 = 20 nM T94119 CA8MV5 44577594 IC50 = 153 nM T94119 C9IXW8 44577638 IC50 = 94 nM T94119 C8A5RT 44577639 IC50 = 21 nM T94119 CNP02V 44577640 IC50 = 26 nM T94119 CT6GN5 44577641 IC50 = 123 nM T94119 CIQR97 44577850 IC50 = 1631 nM T94119 CCG8P9 44577851 IC50 = 11240 nM T94119 CNF47Q 44577852 IC50 = 15280 nM T94119 CLBA40 44577853 IC50 = 783 nM T94119 COU6V7 44577854 IC50 = 605 nM T94119 C8M5FY 44577914 IC50 = 366 nM T94119 C3MGZ9 44577915 IC50 = 1050 nM T94119 CGO09K 44577916 IC50 = 50 nM T94119 CRJ3B7 44577917 IC50 = 155 nM T94119 CTR89C 44577918 IC50 = 7574 nM T94119 CO05YG 44577919 IC50 = 81 nM T94119 CT70WA 44577920 IC50 = 17 nM T94119 C5KXS4 44577921 IC50 = 90 nM T94119 CZ2HI5 44577922 IC50 = 51 nM T94119 CGTU34 44577950 IC50 = 285 nM T94119 CQC50R 44577951 IC50 = 49 nM T94119 C8ZTW2 44577952 IC50 = 230 nM T94119 CIL93G 44577953 IC50 = 357 nM T94119 C8NB5H 44578037 IC50 > 40000 nM T94119 CX9TO2 44578038 IC50 = 19040 nM T94119 C7AHR4 44578039 IC50 > 50000 nM T94119 C13LGI 44578040 IC50 > 50000 nM T94119 CNZ06H 44578074 IC50 > 50000 nM T94119 C41TYA 44578108 IC50 = 74 nM T94119 C2W3SQ 44578109 IC50 = 60 nM T94119 CYM69I 44580064 IC50 = 9 nM T94119 CV09JM 44580065 IC50 = 21 nM T94119 CF37TO 44580066 IC50 = 30 nM T94119 CA0BU6 44580067 IC50 = 245 nM T94119 COQ85J 44580235 IC50 = 12 nM T94119 CD4ER0 44580236 IC50 = 7 nM T94119 CHVQ28 44580237 IC50 = 6 nM T94119 C8N2AF 44580238 IC50 = 103 nM T94119 C40LVX 44580274 IC50 = 231 nM T94119 CO9LD8 44580275 IC50 = 103 nM T94119 C5QWG4 44580276 IC50 = 89 nM T94119 CFZS45 44580277 IC50 = 72 nM T94119 CQ4CR6 44580635 IC50 = 32 nM T94119 CJHK57 44580636 IC50 = 65 nM T94119 CC6M2E 44580684 IC50 = 17 nM T94119 CA3KP5 44580685 IC50 = 43 nM T94119 C40VHS 44580686 IC50 = 14 nM T94119 CXV92J 44580687 IC50 = 29 nM T94119 CG3PH2 44580721 IC50 = 45 nM T94119 CIO46B 44580722 IC50 = 4 nM T94119 CNLS71 44580723 IC50 = 4 nM T94119 C1N0MF 44580724 IC50 = 8 nM T94119 CAHQ76 44580766 IC50 = 39 nM T94119 C2XN6B 44580767 IC50 = 4 nM T94119 CC36YN 44580768 IC50 = 36 nM T94119 CZ56FY 44580769 IC50 = 14 nM T94119 C0L2HO 44593630 IC50 = 139 nM T94119 C2NQ6Z 44593631 IC50 = 16 nM T94119 CY3SV7 44596118 IC50 > 10000 nM T94119 C47FHE 44608747 IC50 < 30 nM T94119 CH6V9F 44608754 IC50 = 6 nM T94119 C0IY9N 44608757 IC50 = 6 nM T94119 C90ITS 44608915 IC50 = 4.3 nM T94119 CZH1P9 44609387 IC50 = 4.4 nM T94119 CNDX48 44609388 IC50 = 5.6 nM T94119 C2ISK4 44610761 IC50 = 47000 nM T94119 CE95RQ 44620964 IC50 = 1.4 nM T94119 CVYJ36 44620965 IC50 = 6.6 nM T94119 CA8BY7 44621440 IC50 < 19952623.15 nM T94119 C5M1FR 44621441 IC50 = 31622776.6 nM T94119 C5LD7E 44621442 IC50 = 12589254.12 nM T94119 CO4GT0 44621447 IC50 = 25118864.32 nM T94119 CUV26H 44621448 IC50 = 7943282.35 nM T94119 CV2MG9 44621449 IC50 = 31622776.6 nM T94119 C24IYW 44621451 IC50 = 25118864.32 nM T94119 C0F9YW 44621452 IC50 = 19952623.15 nM T94119 C0GRD8 44621454 IC50 = 39810717.06 nM T94119 C4YHJ0 44621456 IC50 = 31622776.6 nM T94119 C31VBF 44621458 IC50 = 7943282.35 nM T94119 CZ68MG 45488079 IC50 = 945 nM T94119 CV1U7I 46180604 IC50 = 2.4 nM T94119 CED2B3 46180606 IC50 = 310 nM T94119 CDV85O 46180663 IC50 = 100 nM T94119 CZGB46 46180666 IC50 = 5.2 nM T94119 CAU17V 46202808 IC50 = 79.43 nM T94119 CDA3R9 46220225 IC50 = 11 nM T94119 CM82RF 46239494 IC50 = 9 nM T94119 C7RF5Y 46239967 IC50 = 440 nM T94119 C9Z4HV 46830931 IC50 = 676 nM T94119 CIU7W9 46831535 IC50 = 11 nM T94119 CH59DF 46832094 IC50 > 1000 nM T94119 CD05UP 46832357 IC50 = 292 nM T94119 C94YRI 46853654 IC50 = 15.85 nM T94119 C45JIE 46861590 Ki = 3 nM T94119 CZ3WS1 46861592 IC50 = 0.4 nM T94119 CQ2Y1V 46866705 Ki = 0.122 nM T94119 C63RCG 46870269 IC50 = 12.59 nM T94119 CTQ25M 46871497 IC50 = 63.1 nM T94119 CV96TI 46871579 IC50 < 100 nM T94119 CQB16A 46872415 IC50 > 20000 nM T94119 C3HMQ2 46891474 IC50 = 0.6 nM T94119 CB6Z8P 46892208 IC50 = 5800 nM T94119 CZX46Y 46892342 IC50 = 890 nM T94119 C5FN6I 46892845 IC50 = 510 nM T94119 CQ32BN 46892970 IC50 = 3 nM T94119 COJA32 46892971 Ki = 11 nM T94119 C5QFB3 46893088 IC50 = 320 nM T94119 CS30AI 46893754 IC50 = 4000 nM T94119 CJ0VB4 46932297 IC50 = 330 nM T94119 CF14PE 46947264 IC50 = 77 nM T94119 CV90JU 49764911 IC50 = 10000 nM T94119 COE37N 49778924 IC50 = 20 nM T94119 C7ZK3D 49783923 Ki = 0.07943 nM T94119 CHX76J 49784892 Ki = 37 nM T94119 CA1H8S 49784893 Ki = 130 nM T94119 CP2QD0 49784894 Ki = 2 nM T94119 CTZG05 49784988 Ki = 25 nM T94119 CE9AC5 49785078 Ki = 360 nM T94119 CG2IO7 49785079 Ki = 350 nM T94119 C8EYN4 49785083 Ki = 18 nM T94119 CZI34V 49785167 Ki = 810 nM T94119 CJK65T 49785253 Ki = 56 nM T94119 CXK8F5 49785436 Ki = 2 nM T94119 CWL5C6 49785518 Ki = 6 nM T94119 C3NV0J 49785827 Ki = 9 nM T94119 C0OZM2 49785828 Ki = 27 nM T94119 C1AR4G 49785829 Ki = 5000 nM T94119 CA67CQ 49787183 Ki = 0.23 nM T94119 CIR6Z0 49820690 IC50 < 100 nM T94119 CG74VX 49820826 IC50 = 5.6 nM T94119 CKV2N6 49820977 IC50 = 10 nM T94119 CIO24J 49831132 Ki = 5 nM T94119 C50PCV 49831209 Ki = 1.05 nM T94119 C54OBC 49832773 IC50 = 29 nM T94119 C2G0HN 49832939 IC50 = 2.4 nM T94119 C65WEP 49833295 IC50 = 180 nM T94119 C76XBM 49834039 IC50 = 0.67 nM T94119 CGO57N 49834218 IC50 = 3.5 nM T94119 C90JBE 49834576 Ki = 2 nM T94119 CO2LQ5 49834577 IC50 = 19 nM T94119 C5UR4A 49843944 IC50 = 2020 nM T94119 CS40YB 49853846 IC50 = 400 nM T94119 C7PER0 49853953 IC50 = 69 nM T94119 CU9A8O 49854022 IC50 = 1770 nM T94119 C51QVH 49854023 IC50 = 278 nM T94119 CM4HQ2 49854024 IC50 = 2215 nM T94119 C1LBX3 49854049 IC50 = 70 nM T94119 CVC2H6 49854052 IC50 = 64 nM T94119 CC2X9N 49854121 IC50 = 4290 nM T94119 CAJ58E 49854156 IC50 = 110 nM T94119 CAU39Y 49854158 IC50 = 110 nM T94119 CPK6X3 49854360 IC50 = 700 nM T94119 CQ1TZ6 49854365 IC50 = 1600 nM T94119 CJ5I9X 49854461 IC50 = 910 nM T94119 CDXQ69 49854462 IC50 = 5600 nM T94119 C0ORZ9 49854466 IC50 = 1000 nM T94119 CEC10T 49854573 IC50 = 21 nM T94119 C39KQW 49854679 IC50 = 220 nM T94119 C8VDR2 49854680 IC50 = 230 nM T94119 CN2V8R 49854681 IC50 = 970 nM T94119 CSN96A 49855001 IC50 = 390 nM T94119 CALY90 49855192 IC50 = 3900 nM T94119 CJPE20 49855193 IC50 = 1500 nM T94119 CY8MP7 49867926 IC50 = 43 nM T94119 CR0IA5 49871864 IC50 = 8.8 nM T94119 C13WJZ 49872243 IC50 = 1.4 nM T94119 C5OY7B 49872246 IC50 = 0.8 nM T94119 C2KD5E 49872344 IC50 = 1.3 nM T94119 CV5BF3 49872645 IC50 = 1.3 nM T94119 CN97FO 49872646 IC50 = 0.2 nM T94119 CD6P5R 49872735 IC50 = 1.3 nM T94119 CL64NB 49872737 IC50 = 51 nM T94119 CRNG04 49872831 IC50 = 0.8 nM T94119 CQC8B4 49872835 IC50 = 0.6 nM T94119 CPS3O1 49872924 IC50 = 0.4 nM T94119 CUBX74 49872925 IC50 = 0.2 nM T94119 CAW69U 49872927 IC50 = 0.7 nM T94119 CV1L4P 49873242 IC50 = 4.3 nM T94119 C5BA2V 49873243 IC50 = 12 nM T94119 CSN45W 49873329 IC50 = 1.2 nM T94119 C9CW7X 50908894 IC50 = 6 nM T94119 CJ4L8Y 50938829 Ki = 449 nM T94119 CJG65L 50939078 IC50 = 9 nM T94119 CI8QM1 50939080 Ki = 3 nM T94119 CT0IP3 50939081 Ki = 10 nM T94119 C8JD5T 50939209 IC50 = 17 nM T94119 C54EUL 50939212 Ki = 80 nM T94119 CS7Z6U 50939338 IC50 = 6 nM T94119 CXT23Y 50939344 IC50 = 64 nM T94119 C6GH4K 50939865 IC50 = 85 nM T94119 C2I9PS 50939992 IC50 = 362 nM T94119 C9TUE4 50940108 IC50 = 198 nM T94119 CQ93GK 50940110 IC50 = 47 nM T94119 CG4R5C 50940334 IC50 = 626 nM T94119 C2Q0GE 50990922 Ki = 52 nM T94119 CKY3V1 50990924 Ki = 1.2 nM T94119 C5ZF9W 51003380 IC50 = 5100 nM T94119 CY36EH 51003592 IC50 = 794.33 nM T94119 CPA8N1 51039139 Ki > 10000 nM T94119 C6E9WP 51355057 Ki > 10000 nM T94119 C4QE1V 51355058 IC50 = 4000 nM T94119 CO7M9F 51355343 IC50 > 10000 nM T94119 CJ0KM6 51355344 IC50 = 7300 nM T94119 CT0V8F 51355345 Ki > 10000 nM T94119 C0R8XN 51355348 Ki > 10000 nM T94119 C7KT4Z 51355620 Ki > 10000 nM T94119 CI71WE 51355621 Ki = 5147 nM T94119 CLH35Z 51355622 Ki = 7300 nM T94119 CG7T4H 52913198 IC50 = 12 nM T94119 CYU8K9 52913308 IC50 = 4 nM T94119 CD84MT 52913592 IC50 = 110 nM T94119 C2TLG6 52913931 IC50 = 64 nM T94119 CU1P2L 52940797 IC50 = 2400 nM T94119 C2KI6V 52942202 IC50 = 100000 nM T94119 CDHJ08 52942235 IC50 = 490 nM T94119 C4VCY0 52943258 IC50 = 12000 nM T94119 C1XEV2 52943394 IC50 = 156 nM T94119 CHI0P6 52944356 IC50 = 100000 nM T94119 CU16RS 52944387 IC50 = 3600 nM T94119 CWPC54 52945348 IC50 = 125 nM T94119 C4NLX7 52945630 IC50 = 103 nM T94119 CXD6T8 52945845 IC50 = 800 nM T94119 C7ET6Z 52948010 IC50 = 1200 nM T94119 CV5B2C 52949497 IC50 = 15000 nM T94119 C6LFP7 53209481 IC50 = 5.9 nM T94119 CUJ0D4 53209522 IC50 = 2100 nM T94119 C7B4GC 53232894 IC50 <= 10000 nM T94119 CH1Q5D 53234281 IC50 = 3.5 nM T94119 C45JKN 53234283 IC50 = 3.4 nM T94119 C7I6YV 53234922 IC50 < 250 nM T94119 CVK28S 53235062 IC50 < 0.5 nM T94119 COW61E 53235216 IC50 = 2.6 nM T94119 CWE56X 53235217 IC50 = 1.4 nM T94119 CDXM59 53235451 IC50 = 10.2 nM T94119 CD4ZW8 53240744 IC50 <= 10000 nM T94119 CT8IN1 53242225 IC50 = 890 nM T94119 C73RPF 53250077 IC50 = 430 nM T94119 C2UY0C 53252131 IC50 = 13 nM T94119 C4J9WZ 53307606 IC50 = 1.7 nM T94119 C84YNK 53317325 IC50 = 12000 nM T94119 C58NQJ 53318614 IC50 = 43000 nM T94119 C10YUH 53318615 IC50 = 8900 nM T94119 C24GBF 53319075 IC50 = 49 nM T94119 CFJD70 53319932 IC50 = 40800 nM T94119 C3EJB1 53319933 IC50 = 6500 nM T94119 CJRM64 53322563 IC50 = 11100 nM T94119 CN92LK 53322732 IC50 = 20 nM T94119 C23HAU 53361718 IC50 = 5.9 nM T94119 CM60WQ 53361719 IC50 = 6 nM T94119 CL69DK 53377727 IC50 = 29 nM T94119 C6Q8RC 53378051 IC50 = 3.8 nM T94119 CT43IL 53378053 IC50 = 2.6 nM T94119 CBC63U 53378054 IC50 = 27 nM T94119 CF9D0E 53378155 IC50 = 55 nM T94119 C6OQ4K 53378156 IC50 = 6.3 nM T94119 CPWV36 53378900 IC50 = 12 nM T94119 CP4W1Q 53380858 IC50 = 5011.87 nM T94119 CP0ZU1 53465270 IC50 < 100 nM T94119 CNAY79 53482462 Ki = 0.2 nM T94119 CSV9X2 54579940 IC50 = 11 nM T94119 CN51TL 54579941 IC50 = 4600 nM T94119 C7VZU2 54579942 IC50 = 1300 nM T94119 C4R9JB 54579943 IC50 = 690 nM T94119 CG26HQ 54579944 IC50 = 4600 nM T94119 CC5R3O 54580924 IC50 = 240 nM T94119 C3OIY4 54580925 IC50 = 110 nM T94119 C60TYL 54581049 IC50 = 360 nM T94119 CF2UH5 54581983 IC50 = 71 nM T94119 C23EVN 54582916 IC50 = 140 nM T94119 CT2SV7 54583916 IC50 = 40 nM T94119 CY87EC 54583917 IC50 = 710 nM T94119 C8CPI4 54584859 IC50 = 530 nM T94119 C9TZ2V 54584860 IC50 = 3300 nM T94119 CME81Q 54585830 IC50 = 270 nM T94119 CE4TS9 56589559 IC50 = 1.7 nM T94119 CR24WQ 56595421 IC50 = 34 nM T94119 CJ41GT 56595686 IC50 = 2 nM T94119 C2PN4S 56599298 IC50 = 15 nM T94119 CT64SR 56599306 IC50 = 23 nM T94119 CX37YI 56644424 Ki = 0.46 nM T94119 C3S9XF 56645254 Ki = 0.576 nM T94119 CFUT05 56648675 IC50 = 4.3 nM T94119 C1GAB6 56648677 IC50 = 2.4 nM T94119 CWDF40 56648757 IC50 = 1.5 nM T94119 CE35CB 56648758 IC50 = 5.6 nM T94119 CJO39U 56648759 IC50 = 5 nM T94119 C9DX3J 56649281 IC50 = 144 nM T94119 CNKC90 56654649 IC50 = 28 nM T94119 C94JIT 56832510 Ki = 0.61 nM T94119 C0IJP8 56927258 IC50 = 39.81 nM T94119 CM28GU 56928390 IC50 = 12 nM T94119 C9MJG4 56929824 IC50 = 8 nM T94119 CYFB96 56932203 IC50 = 50.12 nM T94119 CJ9R2C 56932209 IC50 = 6309.57 nM T94119 C8C2FG 56932238 IC50 > 19952.62 nM T94119 CX6Q2K 56932240 IC50 = 79.43 nM T94119 C1G4UV 56933328 IC50 < 50 nM T94119 CO6K5Q 56955953 IC50 = 1134 nM T94119 CAK91L 56955954 IC50 = 18 nM T94119 C8B6JG 56955955 IC50 = 816 nM T94119 CW8B4D 57330208 IC50 = 2.4 nM T94119 C6JMN9 57345685 IC50 = 16 nM T94119 CZ7RE0 57345686 IC50 = 7.9 nM T94119 CA53SC 57351276 Ki = 247 nM T94119 CGU27R 57380079 IC50 < 50 nM T94119 C1X3UP 57390135 IC50 > 1000 nM T94119 CQ6N8D 57390136 IC50 = 220 nM T94119 C6XDC8 57390137 IC50 > 1000 nM T94119 C0S6IG 57390138 IC50 = 10 nM T94119 C2RI4V 57390139 IC50 > 1000 nM T94119 CZ3FU2 57390175 IC50 > 1000 nM T94119 CR2X7O 57390176 IC50 > 1000 nM T94119 C1GVK3 57391362 IC50 = 630 nM T94119 C0PR9J 57391364 IC50 = 63 nM T94119 C6L9HO 57391365 IC50 = 20 nM T94119 C2QX0T 57391366 IC50 = 250 nM T94119 CLQ9J1 57391367 IC50 = 13 nM T94119 C53HZJ 57391915 IC50 > 1000 nM T94119 CO18UJ 57391916 IC50 = 900 nM T94119 CRU8Q0 57391917 IC50 = 510 nM T94119 C13DRO 57391952 IC50 > 1000 nM T94119 CH8UV4 57391962 IC50 = 13 nM T94119 CQ1W0C 57393124 IC50 = 50 nM T94119 CZ0RW2 57393125 IC50 = 630 nM T94119 C3G9VK 57393643 IC50 > 1000 nM T94119 CJX56V 57393644 IC50 = 41 nM T94119 CAND02 57393679 IC50 > 1000 nM T94119 CA93ZE 57394864 IC50 = 160 nM T94119 CF6C2T 57395364 IC50 > 1000 nM T94119 CKE35B 57395365 IC50 = 310 nM T94119 CWL2D6 57395366 IC50 > 1000 nM T94119 CB6L7N 57395397 IC50 > 1000 nM T94119 CJH9S2 57395408 IC50 > 1000 nM T94119 C31MCE 57395409 IC50 = 39 nM T94119 CSP45C 57395410 IC50 = 24 nM T94119 CDG2F3 57396625 IC50 = 40 nM T94119 CD73TE 57396626 IC50 = 800 nM T94119 CQRU75 57396627 IC50 = 130 nM T94119 CI34XH 57396628 IC50 = 40 nM T94119 C92FYK 57397192 IC50 = 32 nM T94119 CBC7N6 57397236 IC50 > 1000 nM T94119 CK01SI 57397253 IC50 = 24 nM T94119 C3Q2ZP 57398390 IC50 = 1300 nM T94119 C56TEZ 57398391 IC50 = 200 nM T94119 CP9Q4U 57398392 IC50 = 250 nM T94119 C0O5KE 57398393 IC50 = 16 nM T94119 C5PI3B 57398894 IC50 > 1000 nM T94119 COTK97 57398895 IC50 > 1000 nM T94119 C3G9HW 57399126 IC50 = 630 nM T94119 CYE09F 57400062 IC50 = 20 nM T94119 CN5PY7 57400063 IC50 = 400 nM T94119 CT0Y7E 57400064 IC50 = 160 nM T94119 C0PZM5 57400579 IC50 > 1000 nM T94119 C9BW8C 57400580 IC50 = 100 nM T94119 C4K2RZ 57400581 IC50 > 1000 nM T94119 C4MW8J 57400582 IC50 > 1000 nM T94119 CGC91E 57400641 IC50 = 22 nM T94119 CM63CS 57401865 IC50 = 16 nM T94119 CG6M4H 57401867 IC50 = 400 nM T94119 CP8FY5 57401868 IC50 = 16 nM T94119 CQ5P4X 57401869 IC50 = 80 nM T94119 C2X8PO 57402386 IC50 = 2500 nM T94119 CNMV98 57402387 IC50 = 59 nM T94119 C06IYP 57402428 IC50 = 230 nM T94119 CF68RN 57403576 IC50 = 1000 nM T94119 CL2R7T 57403577 IC50 = 200 nM T94119 CC5N9R 57403578 IC50 = 100 nM T94119 CZ8M5F 57403579 IC50 = 80 nM T94119 C5NT7R 57403580 IC50 = 31 nM T94119 CHBV63 57403581 IC50 = 3 nM T94119 CAC72X 57403582 IC50 = 1300 nM T94119 CNR95F 57404840 IC50 = 2900 nM T94119 CED47A 57410062 IC50 = 133 nM T94119 C1BVX6 57411134 IC50 = 230 nM T94119 C39JSW 57411135 IC50 = 227 nM T94119 CL8F6Q 57411137 IC50 = 435 nM T94119 CW97FT 57411139 IC50 = 485 nM T94119 CU0R3A 57411250 IC50 = 1555 nM T94119 C6C5TU 57411252 IC50 = 2723 nM T94119 CD0W2I 57411254 IC50 = 178 nM T94119 CW1DA3 57411255 IC50 = 1863 nM T94119 C6U4LO 57411256 IC50 = 134 nM T94119 CP9G7L 57411366 IC50 = 567 nM T94119 CC5DO3 57411369 IC50 = 245 nM T94119 C56RBS 57411372 IC50 = 277 nM T94119 CX9O3T 57411485 IC50 = 1000 nM T94119 CQBM65 57411486 IC50 = 483 nM T94119 CK5QX7 57411488 IC50 = 64 nM T94119 C90LNK 57411715 IC50 = 219 nM T94119 CPXE40 57411716 IC50 = 149 nM T94119 CE6RY5 57411836 IC50 = 127 nM T94119 C5JOX3 57411837 IC50 = 58 nM T94119 C0I5JM 57419280 IC50 > 1000 nM T94119 CNI79K 57427669 IC50 = 7943.28 nM T94119 CT6XL0 57466811 Ki = 470 nM T94119 CWOQ10 57494011 IC50 = 3.1 nM T94119 CRB5P2 57495287 IC50 = 23 nM T94119 C59YAC 57495353 IC50 = 79 nM T94119 CMT9L7 57495355 IC50 = 20 nM T94119 CFIY31 57506723 IC50 = 1.8 nM T94119 CUG89V 57506726 IC50 = 0.48 nM T94119 CVOP28 57506727 IC50 = 6 nM T94119 C48BYL 57506732 IC50 = 2.3 nM T94119 CBZS07 57506734 IC50 = 1.8 nM T94119 CK58VZ 57506735 IC50 = 41 nM T94119 CF1KV7 57506736 IC50 = 12 nM T94119 CBQ5X7 57506737 IC50 = 9.8 nM T94119 C1N8DF 57506739 IC50 = 16 nM T94119 CFH0J4 57506741 IC50 = 2.7 nM T94119 CI30AW 57506743 IC50 = 4.3 nM T94119 CL47BS 57506744 IC50 = 2.3 nM T94119 CJE19S 57523686 IC50 = 5715 nM T94119 CUZ31O 57699545 IC50 < 2000 nM T94119 CV9J7D 57748162 IC50 = 1600 nM T94119 CL57CP 57789333 IC50 = 1090 nM T94119 C81BYH 57798309 IC50 = 310 nM T94119 CZ21KP 57900314 IC50 = 3.9 nM T94119 CC60HE 58008590 IC50 = 0.3 nM T94119 CWE7L8 58119648 IC50 = 665 nM T94119 C4MA7Q 58158259 IC50 < 100 nM T94119 CO20YT 58203712 IC50 = 0.6 nM T94119 C7X0OJ 58203779 IC50 = 1.3 nM T94119 CW1M9X 58203976 IC50 = 3.3 nM T94119 COFN62 58203995 IC50 = 8.4 nM T94119 C16GRS 58204034 IC50 = 8.1 nM T94119 CM62NB 58204076 IC50 < 0.5 nM T94119 CGA01N 58204242 IC50 = 1.1 nM T94119 CVR9Q2 58233988 IC50 = 7.943 nM T94119 CB9AH8 58234990 IC50 = 150 nM T94119 CJ8YI2 58234995 IC50 = 90 nM T94119 CZF3U5 58235016 IC50 = 59 nM T94119 CM0ND7 58235018 IC50 = 59 nM T94119 C25RXY 58235020 IC50 = 61 nM T94119 CAY94U 58235030 IC50 = 76 nM T94119 CAJC03 58235033 IC50 = 44 nM T94119 CN7MZ8 58235039 IC50 = 160 nM T94119 CPW84H 58235041 IC50 = 52 nM T94119 C70CRN 58235043 IC50 = 120 nM T94119 C5SQV3 58235052 IC50 = 73 nM T94119 CEZ4T5 58235053 IC50 = 115 nM T94119 C82LIS 58235061 IC50 = 54 nM T94119 C3SO4E 58235062 IC50 = 62 nM T94119 CZ0SD5 58235073 IC50 = 71 nM T94119 CQP25T 58235077 IC50 = 50 nM T94119 C0LDZ2 58235079 IC50 = 110 nM T94119 C2YG5L 58235088 IC50 = 73 nM T94119 C9N7DV 58329366 IC50 < 100 nM T94119 CWYE70 58346211 IC50 = 27 nM T94119 CVHE56 58532021 IC50 = 5 nM T94119 CZEV29 59146228 IC50 < 100 nM T94119 CJ6R8Q 59251679 IC50 = 100 nM T94119 CRZ5B1 59251991 IC50 = 540 nM T94119 CILJ94 59293648 IC50 = 360 nM T94119 C6A3KL 59293676 IC50 = 3000 nM T94119 CC14ZL 59293709 IC50 = 2000 nM T94119 C0R3TX 59293715 IC50 = 960 nM T94119 C9TVC6 59293721 IC50 = 430 nM T94119 CZ5OV1 59293740 IC50 = 2500 nM T94119 CB2Z4R 59293755 IC50 = 1100 nM T94119 C8AL6C 59293763 IC50 = 690 nM T94119 CUVO13 59362157 Ki = 100 nM T94119 CT3CF1 59477024 IC50 > 5011.87 nM T94119 CF6YB8 59477038 IC50 > 100000 nM T94119 CK3H9O 59477041 IC50 = 1258.93 nM T94119 C7KG5E 59477042 IC50 > 39810.72 nM T94119 C01DZW 59477048 IC50 = 1000 nM T94119 C2X8TY 59548177 Ki = 19 nM T94119 CGRO45 59548196 Ki = 60 nM T94119 CD39AG 59548207 Ki > 10000 nM T94119 C6KP4G 59548220 Ki = 63 nM T94119 CTNU85 59548226 Ki = 110 nM T94119 CLB6N4 59548232 Ki = 5700 nM T94119 CSWV07 59548243 Ki = 34 nM T94119 CMT2R0 59548250 Ki = 240 nM T94119 C3I8NE 59548256 Ki = 51 nM T94119 C8W5HT 59548263 Ki = 310 nM T94119 CT8Q5B 59548274 Ki = 7 nM T94119 CVF1B2 59548283 Ki = 62 nM T94119 CY31EA 59548284 Ki = 30 nM T94119 CO4GT7 59548288 Ki = 0.4 nM T94119 CFR7S8 59548302 Ki = 20 nM T94119 CRM20Z 59548320 Ki = 50 nM T94119 CJE5I4 59548341 Ki = 92 nM T94119 C8O1VS 59548349 Ki = 3 nM T94119 CWC65A 59548356 Ki = 3 nM T94119 CMKP95 59548371 Ki = 7 nM T94119 CC8UV3 59548383 Ki = 70 nM T94119 CD4ET2 59548402 Ki = 130 nM T94119 CES59T 59548403 Ki = 300 nM T94119 CE8P3G 59548407 Ki = 6.1 nM T94119 CO4K2W 59548419 Ki = 1.1 nM T94119 CSDB78 59548424 Ki = 4 nM T94119 C81FCQ 59548431 Ki = 6 nM T94119 CLGY34 59548453 Ki = 15 nM T94119 CBT21W 59548454 Ki = 370 nM T94119 CJT68K 59548460 Ki = 39 nM T94119 C9LFT3 59548462 Ki = 1 nM T94119 CX8C2U 59548480 Ki > 10000 nM T94119 C3TU1N 59605243 IC50 = 4 nM T94119 CW4KI5 59605264 Ki = 2 nM T94119 C7F2UV 59605328 IC50 = 2.74 nM T94119 C1OH9X 59605427 IC50 = 23 nM T94119 CAB24G 59605488 IC50 = 3 nM T94119 C09EWP 59605535 Ki = 0.36 nM T94119 CFCQ97 59605669 IC50 = 39 nM T94119 C7U0JF 59605672 IC50 = 7 nM T94119 C5VP8F 59605730 Ki = 0.8 nM T94119 C5B7OK 59605803 IC50 = 1 nM T94119 C8S0ED 59605870 IC50 = 6 nM T94119 C8R0JT 59606002 IC50 = 5.3 nM T94119 CHO01A 59606100 Ki = 1.8 nM T94119 CW9VH5 59606123 Ki = 12.7 nM T94119 C1N8IZ 59606138 IC50 = 2 nM T94119 CYX9T8 59606142 IC50 = 50 nM T94119 C9MEB6 59606148 Ki = 3.1 nM T94119 C4Y3GL 59609976 IC50 = 125 nM T94119 C1PC0J 59634638 IC50 = 2.8 nM T94119 CP2UY3 59634686 IC50 = 2.9 nM T94119 C1TH2N 59634692 IC50 = 8.3 nM T94119 CPA0L2 59634709 IC50 = 3.6 nM T94119 CBI0M6 59688563 IC50 = 25.12 nM T94119 COFZ83 59753763 IC50 = 270 nM T94119 CUYB59 60148924 IC50 = 800 nM T94119 CM8PD7 60150509 IC50 = 4 nM T94119 C5KD3Z 60154714 Ki > 10000 nM T94119 CS0L4D 60154996 Ki > 10000 nM T94119 C1UI3P 60155086 Ki = 6000 nM T94119 CX08ON 60155087 Ki = 910 nM T94119 CX8J1I 60155265 Ki = 10 nM T94119 CAT40I 60155266 Ki = 4 nM T94119 CD56VA 60155268 Ki = 16 nM T94119 CCQB56 60155375 IC50 = 387 nM T94119 CH5X2S 60155376 IC50 = 456 nM T94119 C74FEN 60155377 IC50 = 1095 nM T94119 CZ6G4B 60155378 IC50 = 352 nM T94119 C10AHQ 60155379 IC50 = 1073 nM T94119 C5FI4P 60155451 Ki = 6 nM T94119 CX9G4U 60155452 Ki = 3 nM T94119 C9Q7DE 60155469 IC50 = 638 nM T94119 CH8UY5 60155470 IC50 = 1418 nM T94119 C3EDY4 60155471 IC50 = 1202 nM T94119 CE0ZX1 60155472 IC50 = 1582 nM T94119 CG90MC 60155473 IC50 = 533 nM T94119 C82PVI 60155474 IC50 = 3389 nM T94119 CX49FT 60155475 IC50 = 2964 nM T94119 CR7EG9 60155538 Ki = 21 nM T94119 CU6YB9 60155539 Ki = 13 nM T94119 CW6N1S 60155552 IC50 = 100 nM T94119 CIB08V 60155553 IC50 = 568 nM T94119 CZE28G 60155554 IC50 = 415 nM T94119 CZD2W7 60155555 IC50 = 546 nM T94119 CO6IU3 60155556 IC50 = 1355 nM T94119 C6HN5O 60155557 IC50 = 437 nM T94119 CMQ9G1 60155638 IC50 = 1020 nM T94119 CG56KT 60155639 IC50 = 539 nM T94119 CBJ65P 60155640 IC50 = 1253 nM T94119 C8OJK0 60155641 IC50 = 340 nM T94119 CT9XJ6 60155642 IC50 = 1186 nM T94119 C5BYQ3 60155643 IC50 = 1032 nM T94119 C57RBF 60155722 IC50 = 743 nM T94119 CU7J6L 60155723 IC50 = 2452 nM T94119 CSZA16 60155724 IC50 = 34 nM T94119 C21DWT 60155725 IC50 = 4389 nM T94119 C12CQU 60155726 IC50 = 1316 nM T94119 CA5TM3 60155805 IC50 = 181 nM T94119 C60RIO 60155806 IC50 = 41 nM T94119 CWC26U 60165513 IC50 = 1.1 nM T94119 C67TFB 60165514 IC50 = 134 nM T94119 CPL1G3 60165805 IC50 = 4.3 nM T94119 C54NOW 66552297 IC50 > 100000 nM T94119 CX4HW1 66552298 IC50 > 100000 nM T94119 CEJ54A 66552343 IC50 = 6309.57 nM T94119 CUQ5Y2 66552345 IC50 > 100000 nM T94119 C5F8ZE 66552346 IC50 > 10000 nM T94119 CHQC56 66552347 IC50 > 100000 nM T94119 CS6BQ0 66552348 IC50 > 100000 nM T94119 CGT2V9 66552407 IC50 > 100000 nM T94119 CIJ3C5 66552408 IC50 = 3162.28 nM T94119 C6ZFI1 66552410 IC50 > 100000 nM T94119 C8S7CM 66552411 IC50 > 25118.86 nM T94119 C9A7IK 66552412 IC50 > 100000 nM T94119 CRC24S 66552467 IC50 > 100000 nM T94119 CHU5V3 66552468 IC50 > 100000 nM T94119 C46POH 66552523 IC50 > 100000 nM T94119 C68LXT 66552524 IC50 > 100000 nM T94119 C91JZL 66553214 IC50 = 2210 nM T94119 CUC7B3 66557964 IC50 = 8.6 nM T94119 C9X2TB 66558056 IC50 = 5.1 nM T94119 C5BP3T 66558242 Ki = 2.5 nM T94119 CLR82P 66558244 Ki = 1.7 nM T94119 CUTG05 66558414 Ki = 1.2 nM T94119 C7FKP2 66575655 IC50 = 11 nM T94119 C1R3SI 66653673 IC50 = 358 nM T94119 CF8BZ7 66677439 IC50 = 4 nM T94119 CQ6U8R 66776828 IC50 <= 10000 nM T94119 CN0RE8 66779813 IC50 = 10 nM T94119 C3IP5D 66779815 IC50 = 16 nM T94119 CH86MR 66779905 IC50 = 63 nM T94119 CX2N6E 66779920 IC50 = 320 nM T94119 C9O4TC 66779989 IC50 = 10 nM T94119 CF2UM8 66780001 IC50 = 500 nM T94119 CHU0C5 66780007 IC50 = 3 nM T94119 CGL4V1 66780016 IC50 = 63 nM T94119 C5F6OA 66780027 IC50 = 2000 nM T94119 C8DN7A 66780034 IC50 = 2500 nM T94119 C4AM6R 66780100 IC50 = 13 nM T94119 CZ5P2N 66780118 IC50 = 2 nM T94119 CREA54 66780266 IC50 = 79 nM T94119 CRCA72 66780292 IC50 = 10 nM T94119 CW2SM6 66780337 IC50 = 2 nM T94119 CU54DY 66780379 IC50 = 40 nM T94119 CQ70YA 66780434 IC50 = 160 nM T94119 C8F9UY 66780515 IC50 = 3 nM T94119 CFH6C2 66780644 IC50 = 250 nM T94119 CTZB46 66780835 IC50 > 790 nM T94119 CEP5A2 66780844 IC50 = 500 nM T94119 C51ARE 66788835 Ki = 0.6 nM T94119 C6C8RD 66802145 IC50 = 790 nM T94119 CW12XO 66882257 IC50 = 2400 nM T94119 C6IO1S 66883557 IC50 = 1470 nM T94119 C1HSE0 67035086 IC50 = 120 nM T94119 C38RGB 67035556 IC50 = 6600 nM T94119 C8HOZ9 67041250 IC50 = 4000 nM T94119 C5E4AJ 67050504 IC50 = 7.6 nM T94119 CMWO25 67061712 IC50 < 0.5 nM T94119 C1K5PQ 67094257 Ki = 630 nM T94119 CJ46YU 67094333 Ki = 890 nM T94119 C0OX5N 67103709 IC50 = 41 nM T94119 C9J2EO 67103712 IC50 = 28 nM T94119 CM4W1Y 67103722 IC50 = 32 nM T94119 C5TYQ3 67103909 IC50 = 12 nM T94119 CVJ49E 67103974 IC50 = 53 nM T94119 C3VFY7 67104025 IC50 = 73 nM T94119 CC07KA 67104052 IC50 = 79 nM T94119 C4Z0HT 67159178 IC50 <= 10000 nM T94119 C7EZW6 67192973 IC50 = 82 nM T94119 C1OXI2 67284515 IC50 = 64 nM T94119 CQHF85 67284779 IC50 = 30 nM T94119 C3K4DG 67285093 IC50 = 72 nM T94119 CYD3P9 67285103 IC50 = 450 nM T94119 CT6BX3 67285457 Ki = 154 nM T94119 CY0C7J 67492428 IC50 = 2 nM T94119 C28DWV 67492561 IC50 = 3 nM T94119 CN2Q1E 67492705 IC50 = 5 nM T94119 CEG3F8 67983123 IC50 = 1200 nM T94119 CA18UP 67983576 IC50 > 9100 nM T94119 C8Z0SM 67983581 IC50 = 500 nM T94119 C2Z4HF 67983896 IC50 = 8500 nM T94119 C26TPD 67983918 IC50 = 820 nM T94119 C25AHY 67984037 IC50 = 7000 nM T94119 C7N4ZS 68034365 IC50 = 820 nM T94119 CC19KE 68041083 IC50 = 3.6 nM T94119 C07EHN 68070485 IC50 < 50 nM T94119 C8I7GC 68293638 IC50 > 10000 nM T94119 C19GYQ 68312763 Ki = 0.78 nM T94119 CUN2V4 68312817 Ki = 2.4 nM T94119 CE43WU 68312934 Ki = 2.8 nM T94119 CM19NS 68312957 Ki = 0.88 nM T94119 CAV08T 68313105 Ki = 0.48 nM T94119 C2K0BV 68313143 Ki = 0.81 nM T94119 CR57TQ 68313151 Ki = 1.9 nM T94119 C7TBV6 68498844 IC50 = 94 nM T94119 COQ61U 68501846 IC50 = 680 nM T94119 C4QT2C 68502605 IC50 = 160 nM T94119 CA4LT5 68502607 IC50 = 950 nM T94119 CO5GZ4 68502623 IC50 = 74 nM T94119 CMS39R 68502742 IC50 = 380 nM T94119 C6OUA7 68502808 IC50 = 450 nM T94119 C09HWK 68502836 IC50 = 27 nM T94119 CI1HJ5 68504925 IC50 > 1000 nM T94119 CAB0C1 68505903 IC50 = 350 nM T94119 C01QHM 68547896 IC50 = 200 nM T94119 C53LRM 70673659 IC50 = 210 nM T94119 C0WIT6 70674249 IC50 = 380 nM T94119 C86YWH 70674360 IC50 = 11 nM T94119 C9CZ5S 70674587 IC50 = 18 nM T94119 C45DBH 70674589 IC50 = 7 nM T94119 C0T7CZ 70674590 IC50 = 6.5 nM T94119 C8MTV6 70674592 IC50 = 4.7 nM T94119 C3F7RY 70675053 IC50 = 3 nM T94119 C3BP8R 70675057 IC50 = 6.6 nM T94119 C4XV9C 70675169 IC50 = 76 nM T94119 CAR46Z 70675172 IC50 = 4.6 nM T94119 C16VLO 70675294 IC50 = 51 nM T94119 C97HZQ 70675296 IC50 = 150 nM T94119 CUV7X5 70675427 IC50 = 35 nM T94119 CN09DI 70675846 IC50 = 168 nM T94119 C6BQE1 70681248 IC50 = 40 nM T94119 CPE36T 70681262 IC50 = 25 nM T94119 CPX41V 70682086 IC50 = 25.12 nM T94119 CQW54O 70682591 Ki = 190 nM T94119 CPV59G 70682592 Ki = 1670 nM T94119 CB3ZN5 70683337 IC50 = 130 nM T94119 C1I5PH 70683338 IC50 = 40 nM T94119 CSM0A6 70684204 IC50 = 6.31 nM T94119 CXD08N 70684690 Ki = 74 nM T94119 C8O2QH 70685440 IC50 = 50 nM T94119 CZG9M1 70685441 IC50 = 79 nM T94119 CH7KO0 70685442 IC50 = 25 nM T94119 C6G4WB 70686339 IC50 > 25118.86 nM T94119 CON8X4 70686340 IC50 = 1584.89 nM T94119 C1ASW4 70686341 IC50 = 12.59 nM T94119 C0PWL5 70686455 IC50 = 1258.93 nM T94119 CN4CR2 70686584 IC50 = 260 nM T94119 C85FWA 70686829 Ki = 19 nM T94119 CQS8G7 70686830 Ki = 220 nM T94119 C8QSD2 70688455 IC50 = 15.85 nM T94119 CFCJ02 70688558 IC50 = 19.95 nM T94119 CSX6I7 70688908 Ki = 210 nM T94119 C5YN6U 70689166 IC50 = 500 nM T94119 C6L4WY 70689639 IC50 = 20 nM T94119 CGT1X2 70690496 IC50 = 199.53 nM T94119 CW3U5J 70690994 Ki = 260 nM T94119 CC6I1Q 70691259 IC50 = 1000 nM T94119 CD3JL4 70691776 IC50 = 31 nM T94119 CDK52M 70692650 IC50 = 794.33 nM T94119 CGQJ68 70692914 IC50 > 1000 nM T94119 C7G5UV 70692915 IC50 = 125.89 nM T94119 C3TM1F 70693128 Ki = 79 nM T94119 C2VAU8 70693129 Ki = 61 nM T94119 C65FHO 70694723 Ki = 8 nM T94119 CPFO83 70694805 IC50 = 794.33 nM T94119 CRNY76 70695188 Ki = 79 nM T94119 C3N5YJ 70695189 Ki = 3620 nM T94119 C75YGN 70695469 IC50 = 50 nM T94119 C61CFG 70696737 IC50 = 25.12 nM T94119 C7KL5X 70696852 IC50 = 3162.28 nM T94119 CRH8E2 71270723 IC50 = 25.12 nM T94119 CWR58A 71270783 IC50 = 158.49 nM T94119 CF9LU4 71270807 IC50 = 19.95 nM T94119 C7FDL2 71270817 IC50 = 15.85 nM T94119 CNR1G9 71270824 IC50 = 125.89 nM T94119 C38LBA 71270831 IC50 = 25.12 nM T94119 CTL6R5 71270836 IC50 = 19.95 nM T94119 CM4LX7 71270848 IC50 > 630.96 nM T94119 C2GWX6 71270906 IC50 > 501.19 nM T94119 CX0DL3 71270910 IC50 = 630.96 nM T94119 C0COW6 71270913 IC50 > 630.96 nM T94119 CB0S8G 71270927 IC50 = 6.31 nM T94119 C24IOW 71270948 IC50 > 630.96 nM T94119 C5BJ2Y 71270957 IC50 > 251.19 nM T94119 C03NFY 71271625 IC50 > 630.96 nM T94119 CL47JU 71271739 IC50 > 398.11 nM T94119 CS5JG6 71271910 IC50 = 100 nM T94119 C4PSK8 71271965 IC50 = 100 nM T94119 CB4N1M 71272066 IC50 > 630.96 nM T94119 CD8E1Y 71272453 IC50 = 25.12 nM T94119 C8EW9V 71272757 IC50 = 158.49 nM T94119 C0LO8I 71272765 IC50 = 79.43 nM T94119 C5A8WF 71449463 IC50 = 4 nM T94119 CWMY48 71450782 IC50 = 111 nM T94119 CNHJ63 71451228 IC50 = 8359 nM T94119 C7V3SO 71452608 IC50 = 139 nM T94119 C6KP3Z 71452609 IC50 < 600 nM T94119 C6W7ZU 71453081 IC50 = 0.6 nM T94119 CR84JX 71453419 Ki = 3 nM T94119 CZQW69 71453554 IC50 > 1000 nM T94119 CZ61FJ 71454160 IC50 = 31622776.6 nM T94119 CZ8Q5P 71454238 Ki = 1.2 nM T94119 C8QIB3 71454374 IC50 = 6 nM T94119 CGD6P2 71456119 IC50 = 3 nM T94119 CYR4J3 71456120 Ki = 3 nM T94119 CYL1G5 71456121 IC50 < 100 nM T94119 CG3OF4 71456597 IC50 = 1.9 nM T94119 CGL8Y4 71457063 IC50 = 6 nM T94119 CDG92F 71457924 IC50 = 14 nM T94119 CPI9J7 71457925 IC50 = 13 nM T94119 C9TAF0 71457926 IC50 = 40 nM T94119 CR14QX 71461548 IC50 = 260 nM T94119 CA6QB4 71461549 IC50 < 100 nM T94119 C3P4RX 71461550 IC50 < 200 nM T94119 CGE64P 71466531 IC50 = 210 nM T94119 CIHT92 71508937 IC50 = 120 nM T94119 CU3EO6 71520393 IC50 = 110 nM T94119 CYC6S1 71520394 IC50 = 2770 nM T94119 C1KMX0 71520395 IC50 = 458 nM T94119 CYK7N8 71520396 IC50 = 1120 nM T94119 CTC0O8 71520397 IC50 = 423 nM T94119 C0UZ3D 71526877 IC50 = 70 nM T94119 CP05SQ 71526878 IC50 = 2200 nM T94119 CZK6X9 71526879 IC50 = 3600 nM T94119 C8QRE4 71526880 IC50 = 1000 nM T94119 CT3QI8 71526881 IC50 = 1200 nM T94119 CO4MY1 71527005 IC50 = 390 nM T94119 CJC64F 71527006 IC50 = 670 nM T94119 C96WZG 71527007 IC50 = 58 nM T94119 CUC7I1 71527008 IC50 = 290 nM T94119 C09WKC 71527009 IC50 = 330 nM T94119 CSPO76 71527716 IC50 > 630.96 nM T94119 CIN7O1 71527842 IC50 > 630.96 nM T94119 CO6CI7 71528725 IC50 = 110 nM T94119 C5U2ZC 71528726 IC50 = 26 nM T94119 CTKO36 71528727 IC50 = 490 nM T94119 C2KF3X 71533728 IC50 = 152 nM T94119 CI7Q4K 71548718 IC50 = 28 nM T94119 CED62L 71548719 IC50 = 27 nM T94119 C4B0KN 71549093 IC50 = 720 nM T94119 C6PRV1 71655831 IC50 = 0.8 nM T94119 CF7R0Y 71682057 IC50 = 11000 nM T94119 CWG8M3 71682651 IC50 = 380 nM T94119 C6UGW3 71682652 IC50 = 4200 nM T94119 C7BX4K 71682653 IC50 = 770 nM T94119 CQX8N3 71682654 IC50 = 3300 nM T94119 CCG6J1 71682807 IC50 > 10000 nM T94119 CS32HB 71716798 IC50 = 251.19 nM T94119 C07GCV 71716799 IC50 > 630.96 nM T94119 CFW01E 71718034 IC50 = 128 nM T94119 C6XKV1 71819134 Ki = 2.3 nM T94119 C95VEJ 71819543 Ki = 0.59 nM T94119 CC3SY4 71819544 Ki = 0.9 nM T94119 CH5R0B 71819545 Ki = 0.88 nM T94119 C7EY1Q 72163951 Ki = 160 nM T94119 CVT76M 72163952 Ki = 490 nM T94119 C9UOH5 72164062 Ki > 10000 nM T94119 CT3X8G 72164184 Ki > 10000 nM T94119 CNX76A 72544842 IC50 = 1258.93 nM T94119 C29KOU 72709209 IC50 > 10000 nM T94119 CT73IW 72709284 IC50 > 10000 nM T94119 C9P1IG 72943510 IC50 = 2841 nM T94119 CVU2J9 72949025 IC50 = 2 nM T94119 CC6KY3 72949203 IC50 = 1 nM T94119 CYGV85 73051332 IC50 = 21 nM T94119 CV4BH5 73051810 IC50 = 21 nM T94119 C7N0AF 73052137 IC50 = 3 nM T94119 CNTD65 73052455 IC50 = 3 nM T94119 C8EI1X 73673707 IC50 = 3.8 nM T94119 CH75QS 73774946 IC50 = 4.4 nM T94119 CBYN18 73977439 IC50 = 15849 nM T94119 C9V1YR 73977449 IC50 = 2512 nM T94119 CXA90D 73977451 IC50 = 2512 nM T94119 CEZ7L2 73977461 IC50 = 794 nM T94119 CD0T9V 74539799 IC50 = 2.8 nM T94119 C16KOS 74539862 IC50 = 3.4 nM T94119 CQ0UM6 74763795 IC50 = 2210 nM T94119 CS71HC 74763798 IC50 = 2770 nM T94119 C5J4EC 76072924 IC50 = 3 nM T94119 CB7Z1L 76285656 EC50 = 1 nM T94119 C38UYZ 76286219 IC50 < 100 nM T94119 CN2MI8 76310247 IC50 > 50000 nM T94119 CKO41J 76310248 IC50 = 367 nM T94119 CEN9Q5 76310249 IC50 = 7600 nM T94119 CJCF67 76310250 IC50 = 14 nM T94119 CIBQ59 76311315 IC50 = 240 nM T94119 C8BD3K 76311316 IC50 = 90 nM T94119 C6F1CR 76311317 IC50 = 440 nM T94119 C7IDU0 76311318 IC50 = 640 nM T94119 CG40TB 76311319 IC50 > 1000 nM T94119 C5WSZ8 76311320 IC50 > 1000 nM T94119 C0M5SE 76311321 IC50 > 1000 nM T94119 CMR07I 76313939 IC50 > 50000 nM T94119 C5P2CJ 76313940 IC50 = 1140 nM T94119 CAV5Q9 76313941 IC50 = 836 nM T94119 CCY5L6 76314906 IC50 > 1000 nM T94119 CE3Z1I 76314907 IC50 = 1550 nM T94119 CFY10G 76314908 IC50 > 1000 nM T94119 C4UHR5 76314909 IC50 = 250 nM T94119 C1B3VO 76314910 IC50 > 1000 nM T94119 CY0Z4U 76314911 IC50 > 1000 nM T94119 CTVO82 76314912 IC50 > 1000 nM T94119 CCWP56 76314913 IC50 > 1000 nM T94119 C0J6PL 76317466 IC50 > 50000 nM T94119 CVW35P 76317467 IC50 > 50000 nM T94119 CZ1T3C 76317468 IC50 > 50000 nM T94119 C4MKN3 76317469 IC50 = 104 nM T94119 C3JA4F 76317470 IC50 = 770 nM T94119 C4XJ5Y 76317471 IC50 = 565 nM T94119 C3SIE7 76318525 IC50 > 1000 nM T94119 CU6G7L 76318526 IC50 > 1000 nM T94119 CC3Z2U 76318527 IC50 = 2000 nM T94119 C8E4GI 76321204 IC50 = 24 nM T94119 CF4OI8 76321205 IC50 = 1900 nM T94119 CR61ZP 76322185 IC50 > 1000 nM T94119 C5LT0B 76322186 IC50 > 1000 nM T94119 C19SKA 76322187 IC50 > 1000 nM T94119 CDG8V4 76324821 IC50 = 8 nM T94119 CJW39V 76324822 IC50 > 50000 nM T94119 C2BFA1 76324823 IC50 = 18 nM T94119 C1HFI9 76325446 IC50 = 430 nM T94119 C7IFD5 76325803 IC50 > 1000 nM T94119 C2NK4S 76325804 IC50 > 1000 nM T94119 COJ6P9 76325805 IC50 > 1000 nM T94119 C2AJ6T 76325806 IC50 > 1000 nM T94119 C4A8XZ 76328376 IC50 = 5280 nM T94119 C8S2IL 76329389 IC50 > 1000 nM T94119 CAEW42 76329390 IC50 > 1000 nM T94119 CMC32D 76329391 IC50 > 1000 nM T94119 CAZ9Q2 76329392 IC50 > 1000 nM T94119 C06ZQJ 76329393 IC50 = 3350 nM T94119 CYR0G6 76332050 IC50 = 150 nM T94119 C4MID5 76332051 IC50 = 26500 nM T94119 C70WJE 76332052 IC50 = 134 nM T94119 CE6BI0 76332666 IC50 = 63 nM T94119 CKG1E0 76333034 IC50 = 200 nM T94119 C6D4RU 76333035 IC50 > 1000 nM T94119 CSAT72 76333036 IC50 > 1000 nM T94119 C1JRO2 76333037 IC50 > 1000 nM T94119 C8TNI0 76333038 IC50 > 1000 nM T94119 C69ATM 76335666 IC50 > 50000 nM T94119 C0SI4C 76335667 IC50 > 50000 nM T94119 C31NEK 76335668 IC50 = 687 nM T94119 CL6BV5 76335669 IC50 = 11130 nM T94119 C73KJD 76335670 IC50 = 77 nM T94119 CP2UC5 76336660 IC50 > 1000 nM T94119 C79JAI 76336661 IC50 = 150 nM T94119 C2JTH8 77107528 IC50 = 1.9 nM T94119 C42HDP 77107927 IC50 = 4.1 nM T94119 C04SRC 77147259 IC50 = 3225 nM T94119 C9I7TY 78319187 IC50 = 12589.25 nM T94119 C24LQH 78320362 IC50 = 4 nM T94119 C9T8KF 78320671 IC50 < 3 nM T94119 CI2YN8 78320672 IC50 < 3 nM T94119 CI6K4J 78320673 IC50 = 52 nM T94119 COFJ16 78320996 IC50 = 76 nM T94119 CMU5P2 78321310 IC50 = 14 nM T94119 CE13AJ 78321314 IC50 = 11 nM T94119 CSP2H4 78321635 IC50 = 8 nM T94119 CWA0B1 78322567 IC50 = 12 nM T94119 CH6P9D 78322877 IC50 = 43 nM T94119 C4IW9V 78323193 IC50 = 23 nM T94119 CD1JC8 78324443 IC50 = 5 nM T94119 C04IKP 86268622 IC50 = 2.5 nM T94119 C5P3RO 86647783 IC50 = 620 nM T94119 CP7HJ2 86666761 IC50 = 99 nM T94119 CD6XP5 86677746 IC50 = 11 nM T94119 CDXM47 86677874 IC50 < 1 nM T94119 CP3W1B 86695297 IC50 = 15 nM T94119 CA17UE 86732669 IC50 = 9 nM T94119 C2PCS7 87061302 IC50 = 223 nM T94119 CI8X3C 87150169 IC50 = 12589.25 nM T94119 CV6PI8 87562294 IC50 = 316.23 nM T94119 CN4B6P 88536250 IC50 = 5.3 nM T94119 C1HB3F 89051931 IC50 = 8.2 nM T94119 CY64GN 89420800 IC50 = 1.9 nM T94119 C61SCX 89493851 IC50 = 4.9 nM T94119 C1LU3X 89493904 IC50 = 29 nM T94119 CTE1L0 89517065 IC50 = 9 nM T94119 C56KSC 89517226 IC50 = 36 nM T94119 CN5Y9A 90064110 IC50 = 16 nM T94119 C7FP2M 90064111 IC50 = 5 nM T94119 CQE9C3 90158083 IC50 = 8330 nM T94119 C9IOQ0 90158408 IC50 = 45 nM T94119 C9JAI2 90166620 IC50 = 572 nM T94119 C49XDA 90166847 IC50 = 190 nM T94119 CC4M6F 90168602 IC50 = 35 nM T94119 C5LK7G 90168751 IC50 = 1290 nM T94119 CF03DW 90168772 IC50 = 24 nM T94119 CM6J9K 90168778 IC50 = 16 nM T94119 CVF37R 90168935 IC50 = 187 nM T94119 C28WQY 90431726 IC50 = 30 nM T94119 C08UWK 90665816 IC50 = 630 nM T94119 CMWB58 91757958 IC50 <= 10000 nM T94119 C3Y0DS 91801158 IC50 = 59 nM T94119 C2OG7F 91820679 IC50 = 0.7 nM T94119 CAS7W6 91864650 IC50 = 880 nM T94119 C1QJ3K 117815397 IC50 = 4200 nM T94119 CLA03N 117965586 IC50 = 2 nM T94119 C34FKB 118025462 IC50 = 4 nM T94119 CUQS80 118025552 IC50 = 13 nM T94119 C1KGB4 118025559 IC50 = 1830 nM T94119 CDF6L7 118025606 IC50 = 1340 nM T94119 CGX1T6 118025676 IC50 = 61 nM T94119 C1IL8Q 118025680 IC50 = 9 nM T94119 C79ZBM 118025723 IC50 = 33 nM T94119 C6HO9P 118025760 IC50 = 8 nM T94119 CM4Z5V 118025790 IC50 = 2790 nM T94119 CX4W9A 118025823 IC50 = 35 nM T94119 C3FG4U 118025830 IC50 = 32 nM T94119 CM3JO2 118025835 IC50 = 155 nM T94119 CKR9G1 118025928 IC50 = 3 nM T94119 C5TQU3 118025943 IC50 = 8 nM T94119 C68YAU 118026010 IC50 = 172 nM T94119 C14WCU 118131317 IC50 < 10 nM T94119 CE42ID 118165924 IC50 = 0.04 nM T94119 C67VQE 118341819 IC50 > 10000 nM T94119 CC9P5H 118341835 IC50 > 10000 nM T94119 CUMA23 118341844 IC50 = 270 nM T94119 C3IP9X 118341852 IC50 > 10000 nM T94119 C6TI0Z 118341865 IC50 > 10000 nM T94119 C4U7NC 118341870 IC50 > 10000 nM T94119 CVL03K 118341884 IC50 > 10000 nM T94119 CPZN96 118341923 IC50 > 10000 nM T94119 C9E3DU 118341927 IC50 > 10000 nM T94119 CVN87P 118433737 IC50 = 2.7 nM T94119 C8W1RN 118445922 IC50 = 3 nM T94119 CQF1V4 118446049 IC50 = 63 nM T94119 CVYK24 118556943 IC50 = 62 nM T94119 CJQ92T 118572891 IC50 = 10 nM T94119 C2U3BQ 118627731 IC50 = 0.1 nM T94119 CS5C8W 118684133 IC50 = 4.1 nM T94119 CRX24W 118709077 IC50 = 110 nM T94119 CV2EJ7 118709081 IC50 = 85 nM T94119 CZ41AQ 118709092 IC50 = 400 nM T94119 CR6ML1 118709578 IC50 = 51 nM T94119 C0OH7I 118709579 IC50 = 230 nM T94119 C73YIO 118709582 IC50 = 45 nM T94119 CGWX02 118709583 IC50 = 32 nM T94119 CB53EU 118728320 IC50 > 50000 nM T94119 C6KJL1 118728321 IC50 = 42618 nM T94119 CKJ3S6 118728322 IC50 > 50000 nM T94119 CT0L3Y 118728325 IC50 > 50000 nM T94119 CHS2E4 118728326 IC50 > 50000 nM T94119 CRUP47 118728328 IC50 = 47763 nM T94119 CQR41G 118728330 IC50 = 39842 nM T94119 CN4Q9R 118728332 IC50 = 34624 nM T94119 CDI10F 118728336 IC50 > 50000 nM T94119 CHT6K9 118728811 Ki > 4000 nM T94119 CUA3Y2 118728812 Ki > 4000 nM T94119 CDQ78G 118728813 Ki = 3100 nM T94119 CZ6XL7 118728814 Ki = 180 nM T94119 CMO67K 118728815 Ki > 4000 nM T94119 CR2M0Q 118728816 Ki > 4000 nM T94119 C62SCL 118728817 Ki > 4000 nM T94119 CSB30C 118728819 Ki = 1900 nM T94119 CV7XU8 118728820 Ki = 1600 nM T94119 C3J1EX 118728821 Ki > 4000 nM T94119 CIWB78 118728822 Ki > 4000 nM T94119 CP18SE 118728823 Ki > 4000 nM T94119 CM42CA 118728824 Ki = 2500 nM T94119 C9Q7CL 118728825 Ki = 1200 nM T94119 CCR3S0 118728826 Ki = 3300 nM T94119 CB1WC5 118729946 IC50 = 2.5 nM T94119 CQ4G9M 118729947 IC50 = 1.7 nM T94119 C43IPJ 118729948 IC50 = 4 nM T94119 C3I9CQ 118729949 IC50 = 1.4 nM T94119 CZQ17M 118729950 IC50 = 1.2 nM T94119 C3G1ZP 118729951 IC50 = 3.1 nM T94119 CY60FC 118730033 IC50 > 50000 nM T94119 CN3B4U 118730711 IC50 = 22 nM T94119 C0IL3N 118730712 IC50 = 23 nM T94119 C3CH1A 118730713 IC50 = 20 nM T94119 CHX5L9 118730714 IC50 = 14 nM T94119 CNJ32C 118730715 IC50 = 80 nM T94119 C1MKB3 118730716 IC50 = 27 nM T94119 C81RJA 118730717 IC50 = 160 nM T94119 CFZ16R 118737301 IC50 <= 10000 nM T94119 C27CPQ 118737302 IC50 <= 10000 nM T94119 C59VXA 118737303 IC50 <= 10000 nM T94119 CGO1N4 118737304 IC50 <= 10000 nM T94119 CS85FM 118737305 IC50 <= 10000 nM T94119 C8UCO1 118737306 IC50 <= 10000 nM T94119 CR0BZ2 118737307 IC50 <= 10000 nM T94119 C3N4DJ 118737308 IC50 <= 10000 nM T94119 CGY5B1 118737309 IC50 <= 10000 nM T94119 CFN12W 121445751 IC50 = 25.8 nM T94119 CVU7P1 121445752 IC50 = 0.6 nM T94119 C2UDS6 121445784 IC50 = 6 nM T94119 C04NDW 121445810 IC50 = 17.4 nM T94119 CM4Y3Z 121483558 IC50 = 309 nM T94119 C81IFQ 122163152 IC50 = 1840 nM T94119 C2VGD5 122178120 IC50 = 13.3 nM T94119 C24XUZ 122178124 IC50 = 3.1 nM T94119 CN5AB3 122179486 IC50 = 10 nM T94119 CLEK13 122179487 IC50 = 4 nM T94119 C0OW8H 122179490 IC50 = 44 nM T94119 C0VD5F 122179491 IC50 = 63.1 nM T94119 CQ87FB 122179492 IC50 = 199 nM T94119 CBJ29X 122179493 IC50 = 2000 nM T94119 CA5N1B 122179494 IC50 = 20 nM T94119 CSTE64 122179689 IC50 = 220 nM T94119 CE2FM7 122179690 IC50 = 470 nM T94119 CZJ31R 122179691 IC50 = 270 nM T94119 CBOU30 122179692 IC50 = 470 nM T94119 CKWC74 122179693 IC50 = 810 nM T94119 C4CX7Z 122179694 IC50 = 710 nM T94119 C48LYC 122179695 IC50 = 1100 nM T94119 C3D5QM 122179696 IC50 = 240 nM T94119 CW3DM7 122179697 IC50 = 600 nM T94119 C6I3PB 122179698 IC50 > 10000 nM T94119 CCU6A4 122179699 IC50 = 570 nM T94119 C7WMC3 122179700 IC50 = 470 nM T94119 C86NOQ 122179701 IC50 = 550 nM T94119 CAHY19 122179702 IC50 = 460 nM T94119 C3O7CM 122179703 IC50 = 1500 nM T94119 CK2R4X 122179704 IC50 = 410 nM T94119 CG96HD 122179705 IC50 = 900 nM T94119 C1PK9L 122179706 IC50 = 470 nM T94119 CEB69W 122179707 IC50 = 1000 nM T94119 CK97EL 122179708 IC50 = 500 nM T94119 C0ZA4C 122179709 IC50 = 640 nM T94119 CU93YJ 122179710 IC50 = 450 nM T94119 C0KTH8 122179711 IC50 = 150 nM T94119 CN9I1C 122179712 IC50 = 530 nM T94119 C65OGI 122179713 IC50 = 300 nM T94119 C92AZK 122179714 IC50 = 140 nM T94119 CWL43Z 122179715 IC50 > 10000 nM T94119 C50VNH 122179716 IC50 > 10000 nM T94119 COW37C 122179717 IC50 > 10000 nM T94119 CG5N9E 122179718 IC50 = 220 nM T94119 CB14FW 122179719 IC50 = 270 nM T94119 CHZ3S1 122179720 IC50 = 470 nM T94119 CEG8Y6 122179721 IC50 = 30 nM T94119 CG5P3J 122179722 IC50 = 1700 nM T94119 CZH3T1 122179723 IC50 = 480 nM T94119 C10FGR 122179724 IC50 = 1800 nM T94119 CEFS13 122180793 IC50 = 14570 nM T94119 CFZ2E1 122180794 IC50 = 20120 nM T94119 C5YKG7 122180795 IC50 = 71350 nM T94119 C9ID7U 122180796 IC50 = 56890 nM T94119 C08XOC 122180839 IC50 = 120000 nM T94119 C2HM6P 122180840 IC50 = 154780 nM T94119 CT9Y6U 122180841 IC50 = 3550 nM T94119 C6FOM0 122180842 IC50 = 2740 nM T94119 COX90L 122180843 IC50 = 1810 nM T94119 CP40RU 122180844 IC50 = 3970 nM T94119 CC0EK9 122180845 IC50 = 2610 nM T94119 CS85CU 122181413 IC50 = 20 nM T94119 CQS67B 122181416 IC50 = 17 nM T94119 C58XRY 122184465 IC50 = 3981.07 nM T94119 C16ALM 122184466 IC50 = 1995.26 nM T94119 CIX19J 122184467 IC50 = 6309.57 nM T94119 CDZY02 122184468 IC50 = 63095.73 nM T94119 CTH70U 122184469 IC50 = 12589.25 nM T94119 C9ZXR7 122184470 IC50 = 6309.57 nM T94119 CNJ9Z4 122184471 IC50 = 12589.25 nM T94119 CS41EG 122184473 IC50 = 1258.93 nM T94119 CZ36GL 122184474 IC50 = 1000 nM T94119 CU4ZT6 122184475 IC50 = 12589.25 nM T94119 C3H9PR 122184476 IC50 = 1995.26 nM T94119 CU40TW 122184477 IC50 = 6309.57 nM T94119 CAMD31 122184479 IC50 = 63095.73 nM T94119 C1F9RK 122184480 IC50 = 1258.93 nM T94119 C7XW1K 122184481 IC50 = 79432.82 nM T94119 CRUX54 122184482 IC50 = 50118.72 nM T94119 CQ7W0P 122184526 IC50 = 7943.28 nM T94119 CA5YB2 122184529 IC50 = 12589.25 nM T94119 C64YPH 122184530 IC50 = 25118.86 nM T94119 C4AGX5 122184531 IC50 = 19952.62 nM T94119 CQL4K5 122184532 IC50 = 12589.25 nM T94119 CRKV74 122184533 IC50 = 19952.62 nM T94119 CX14YD 122184534 IC50 = 3981.07 nM T94119 CM6A4S 122184535 IC50 = 19952.62 nM T94119 CF86YS 122184536 IC50 = 19952.62 nM T94119 CH08SN 122184537 IC50 = 5011.87 nM T94119 CYRH97 122184538 IC50 = 10000 nM T94119 CD4W0Z 122184539 IC50 > 199526.23 nM T94119 CH8Y3Q 122184540 IC50 = 100000 nM T94119 CDA85R 122184541 IC50 > 199526.23 nM T94119 CF36XJ 122184542 IC50 > 199526.23 nM T94119 CQ6O7H 122184543 IC50 > 199526.23 nM T94119 CS4MN0 122184544 IC50 > 79432.82 nM T94119 CKT74G 122185265 IC50 = 16 nM T94119 CJ6C1O 122185267 IC50 = 12 nM T94119 CK9VY5 122197304 IC50 < 50 nM T94119 CGW35U 122387497 IC50 > 1000 nM T94119 C38BML 122387499 IC50 > 1000 nM T94119 CCW0M1 122387500 IC50 = 553 nM T94119 CKA90Y 122387501 IC50 = 348 nM T94119 CH4LC6 122387502 IC50 = 271 nM T94119 C8OC3E 122387504 IC50 = 674 nM T94119 C34AHY 122387505 IC50 = 722 nM T94119 CUG1T6 122387506 IC50 = 311 nM T94119 CE7K5C 122387507 IC50 = 683 nM T94119 C4HL3N 122387508 IC50 = 474 nM T94119 CA7L3S 122387509 IC50 = 489 nM T94119 CR9NF3 122542400 IC50 = 1.4 nM T94119 CMG21L 122705987 IC50 = 8500 nM T94119 CW5EK9 122705988 IC50 = 640 nM T94119 CPTY78 124518210 IC50 = 2.5 nM T94119 C1N6YP 126480569 IC50 = 110 nM T94119 CE52HC 126480570 IC50 = 90 nM T94119 CPW54V 126480574 IC50 = 50 nM T94119 CVJ3Q5 127025094 IC50 > 1000 nM T94119 C98DKI 127025346 IC50 = 19 nM T94119 CBXJ67 127025628 IC50 = 14 nM T94119 CSV3R7 127029064 IC50 = 50 nM T94119 CQTG79 127029604 IC50 > 1000 nM T94119 C47BCU 127030580 IC50 = 740 nM T94119 CZHT45 127031017 IC50 = 1570 nM T94119 CU0F4R 127031332 IC50 = 340 nM T94119 C2IN4Q 127031333 IC50 = 50000 nM T94119 CS12RU 127031435 IC50 = 12.4 nM T94119 CGU4H3 127031891 IC50 = 33 nM T94119 CGKR53 127032915 IC50 = 2075 nM T94119 CYSN74 127034047 IC50 = 3700 nM T94119 C41YQI 127035981 IC50 > 5000 nM T94119 C2O4RK 127038523 IC50 = 2600 nM T94119 CO27IE 127038894 IC50 = 10000 nM T94119 C72NPR 127039226 IC50 = 4500 nM T94119 CL0ZU8 127040691 IC50 = 2700 nM T94119 CB0G7Z 127040692 IC50 = 10000 nM T94119 C3ZXT2 127040693 IC50 = 9000 nM T94119 CY6NM3 127040694 IC50 > 10000 nM T94119 CLUK47 127042289 IC50 = 12000 nM T94119 C05MRE 127042767 IC50 = 4800 nM T94119 C4L9TC 127042949 IC50 = 3700 nM T94119 CG8DA9 127045861 IC50 = 505 nM T94119 CVF8Z9 127045862 IC50 = 7.3 nM T94119 CH68NT 127046076 IC50 = 149 nM T94119 CA2XD5 127046077 IC50 = 221 nM T94119 COJ68G 127046117 IC50 = 13 nM T94119 C34REM 127046317 IC50 = 11 nM T94119 CC4ND8 127046862 IC50 = 271 nM T94119 CY2P1X 127047138 IC50 = 11 nM T94119 CZ2R0C 127047140 IC50 = 10 nM T94119 CT89GI 127047683 IC50 = 14 nM T94119 C7D0FN 127047685 IC50 = 7 nM T94119 CN94CQ 127047797 IC50 = 9 nM T94119 C5OE2H 127053611 IC50 = 71 nM T94119 CN9XL1 129262531 IC50 = 1 nM T94119 C92EMK 129395626 IC50 = 3.6 nM T94119 CW7A5X 129626595 IC50 = 31.62 nM T94119 CGIT40 129896911 IC50 = 16 nM T94119 C18NHD 130302549 IC50 <= 10000 nM T94119 CL13RZ 130302558 IC50 <= 10000 nM T94119 CF5JZ3 130302563 IC50 <= 10000 nM T94119 CD46EL 130302605 IC50 <= 10000 nM T94119 CNI8M6 130302620 IC50 <= 10000 nM T94119 CI6WN9 130302651 IC50 <= 10000 nM T94119 C5ZP0L 130302658 IC50 <= 10000 nM T94119 CW61SG 130302663 IC50 <= 10000 nM T94119 CB27ZG 130302668 IC50 <= 10000 nM T94119 C5VYM6 130302674 IC50 <= 10000 nM T94119 C0FQR2 130302675 IC50 <= 10000 nM T94119 CB34HQ 130302676 IC50 <= 10000 nM T94119 CQR1I8 130302685 IC50 <= 10000 nM T94119 C17DZF 130302698 IC50 <= 10000 nM T94119 CBC6W7 130302701 IC50 <= 10000 nM T94119 CBT21G 130302702 IC50 <= 10000 nM T94119 CDZ45O 130302703 IC50 <= 10000 nM T94119 C2GWU8 130302709 IC50 <= 10000 nM T94119 CV3M6Y 130302710 IC50 <= 10000 nM T94119 C39UQN 130302731 IC50 <= 10000 nM T94119 CL9O8X 130302732 IC50 <= 10000 nM T94119 CL69GM 130302740 IC50 <= 10000 nM T94119 CH8YK9 130302741 IC50 <= 10000 nM T94119 CQR2W9 130302781 IC50 <= 10000 nM T94119 C9HC8A 130302803 IC50 <= 10000 nM T94119 CIK25W 130302809 IC50 <= 10000 nM T94119 CI08PF 130332501 IC50 <= 10000 nM T94119 C1H4UT 130332505 IC50 <= 10000 nM T94119 CZPI64 130332579 IC50 <= 10000 nM T94119 CDS9F3 130332582 IC50 <= 10000 nM T94119 C3G0HF 130332585 IC50 <= 10000 nM T94119 CX13UC 130332620 IC50 <= 10000 nM T94119 CED6F3 130332657 IC50 <= 10000 nM T94119 CRG3I4 130362847 IC50 = 0.8 nM T94119 C8W2EJ 130362892 IC50 = 5.2 nM T94119 C3YFV8 130362899 IC50 = 1.8 nM T94119 CP5D7R 130362915 IC50 = 0.4 nM T94119 CUP5N0 130363024 IC50 = 0.6 nM T94119 CD1PV2 130363056 IC50 = 3.5 nM T94119 CKTL52 130363065 IC50 = 2.5 nM T94119 CR8S9K 130363066 IC50 = 5 nM T94119 CJ3Y7M 130363067 IC50 = 7 nM T94119 C19CXK 130363082 IC50 = 1.2 nM T94119 COS6W5 130363083 IC50 = 56 nM T94119 CO1YL7 130363101 IC50 = 24 nM T94119 CE1YZ2 130363102 IC50 = 2.4 nM T94119 CBN3D6 130363112 IC50 = 1 nM T94119 C3QBL4 130363125 IC50 = 0.3 nM T94119 C53JWU 130363129 IC50 = 1.9 nM T94119 C3SK4J 130363145 IC50 = 72 nM T94119 CX8D6O 130363152 IC50 = 3 nM T94119 CK91CJ 130363160 IC50 = 105 nM T94119 C0A2YT 130363168 IC50 = 1 nM T94119 C7E6XI 130363172 IC50 = 0.5 nM T94119 C7JP0R 130363201 IC50 = 3.3 nM T94119 C76YRN 130363211 IC50 = 3 nM T94119 C3Q7LT 130363215 IC50 = 0.9 nM T94119 C7OPB5 130363224 IC50 = 1.9 nM T94119 C64XBS 130363239 IC50 = 98 nM T94119 CN75CD 130363275 IC50 = 4.8 nM T94119 CYTF09 130363280 IC50 = 31 nM T94119 CLAB53 130363290 IC50 = 140 nM T94119 CFI60X 130363298 IC50 = 1.1 nM T94119 C3V9DW 130363308 IC50 > 150 nM T94119 CNO3U9 130363327 IC50 = 5 nM T94119 COKX96 130363382 IC50 = 1 nM T94119 CJO36T 130363391 IC50 = 2 nM T94119 CFXC13 130363397 IC50 = 0.4 nM T94119 C0WS3I 130363410 IC50 = 9 nM T94119 C60KGA 130363411 IC50 = 1.1 nM T94119 C31RSQ 130363418 IC50 = 2 nM T94119 CTN8C0 130363443 IC50 = 1.4 nM T94119 CD54NU 130363457 IC50 = 5 nM T94119 C3PB1V 130363463 IC50 = 4 nM T94119 CNFH51 130363544 IC50 = 0.8 nM T94119 C65ZDT 130363548 IC50 = 5 nM T94119 CULX27 130363568 IC50 = 30 nM T94119 COK9T6 130363592 IC50 = 33 nM T94119 C6CIJ2 130363602 IC50 = 1.5 nM T94119 CFN3Z5 130363612 IC50 = 6 nM T94119 CMX9O5 130363616 IC50 = 5.5 nM T94119 C6H9BS 130363645 IC50 = 2.1 nM T94119 COPI97 130363656 IC50 = 5.5 nM T94119 C0G9LM 130363659 IC50 = 2 nM T94119 COWE45 130363737 IC50 < 0.3 nM T94119 CAK3T1 130363738 IC50 = 2 nM T94119 CR8G9C 130363746 IC50 = 2 nM T94119 C47CAY 130421765 IC50 = 794.33 nM T94119 C84YKI 130422161 IC50 = 398.11 nM T94119 CK68CA 130453737 IC50 = 730 nM T94119 CDE7T3 132005217 IC50 = 120 nM T94119 CL26YS 132005219 IC50 = 96 nM T94119 CP32GB 132005220 IC50 = 29 nM T94119 CG1NC4 132005221 IC50 = 2600 nM T94119 C0UV2M 132005224 IC50 = 41 nM T94119 CUN18W 132005225 IC50 = 2 nM T94119 CD84OI 132005228 IC50 = 1.5 nM T94119 C9VDI0 132005229 IC50 = 230 nM T94119 CB1Z7P 132005231 IC50 = 440 nM T94119 C7ASP9 132005246 IC50 = 1.7 nM T94119 C8VE6T 132005248 IC50 = 51 nM T94119 C7LCW1 132005249 IC50 = 76 nM T94119 C5W9LN 132005323 IC50 = 20 nM T94119 CQ6GO2 132005326 IC50 = 39 nM T94119 C1XUW7 132209432 IC50 = 4.7 nM T94119 CPL60M 132209468 IC50 = 0.6 nM T94119 C6Y4CH 132209868 IC50 = 4 nM T94119 C58NEJ 132209870 IC50 = 19 nM T94119 CIL1Q3 132209885 IC50 = 6.4 nM T94119 CP7N3I 132209920 IC50 = 3 nM T94119 C4M8WN 132209922 IC50 = 1.3 nM T94119 CJ83PK 132209926 IC50 = 3.9 nM T94119 CJ5FI1 132209935 IC50 = 11 nM T94119 CHQP87 132209952 IC50 = 100 nM T94119 C6JGE1 132209957 IC50 = 1.7 nM T94119 C45NEF 132209959 IC50 = 5.5 nM T94119 CZFO16 132209976 IC50 = 1.2 nM T94119 CI6P5H 132209981 IC50 = 6 nM T94119 CCK6E1 132209985 IC50 = 10 nM T94119 COK4X3 132210002 IC50 = 0.9 nM T94119 CTG6C8 132210009 IC50 = 2 nM T94119 C3CFB2 132210012 IC50 = 4.5 nM T94119 CS4V6U 132210025 IC50 = 0.9 nM T94119 CM9P1H 132210051 IC50 = 424 nM T94119 C16HBK 132210068 IC50 = 1.3 nM T94119 CFI23B 132210082 IC50 = 0.5 nM T94119 C02QSJ 132210090 IC50 = 16 nM T94119 C9Q0ZW 132210105 IC50 = 16 nM T94119 CH8DP7 132220479 IC50 < 0.1 nM T94119 C6NWY1 132220480 IC50 = 1 nM T94119 CD7X5S 132220481 IC50 = 2.2 nM T94119 CRC14V 132220484 IC50 = 1.5 nM T94119 C4Q5LF 132471857 IC50 = 7 nM T94119 CJE34F 132597748 IC50 = 18.5 nM T94119 CCV46G 132606879 IC50 = 3.981 nM T94119 C6PWX2 134129963 IC50 = 66 nM T94119 CV2PK1 134129977 IC50 = 100 nM T94119 CSWZ68 134130018 IC50 = 61 nM T94119 CBR3Z9 134130128 IC50 = 88 nM T94119 CM51SI 134130327 IC50 = 55 nM T94119 CLO3M4 134130336 IC50 = 470 nM T94119 CS9Q7P 134130420 IC50 = 575 nM T94119 C0WEA6 134130582 IC50 = 60 nM T94119 C2X1BY 134130678 IC50 = 150 nM T94119 C97JFV 134131108 IC50 = 68 nM T94119 C1LZP4 134131157 IC50 = 100 nM T94119 COI4W0 134131210 IC50 > 1000 nM T94119 C54IJX 134131348 IC50 = 170 nM T94119 C5M6BU 134131349 IC50 = 350 nM T94119 CH17GQ 134131392 IC50 = 130 nM T94119 CIYZ86 134131408 IC50 = 658 nM T94119 C9NYX3 134131539 IC50 = 370 nM T94119 CFG90E 134132909 IC50 = 256 nM T94119 CI49TK 134133218 IC50 = 1.6 nM T94119 C4YNH0 134134126 IC50 = 28 nM T94119 C0EK8P 134134680 IC50 = 11 nM T94119 CU9VC6 134136072 IC50 = 47 nM T94119 CS73WF 134136130 IC50 = 370 nM T94119 C0A1UM 134138053 IC50 = 10 nM T94119 C6OGM2 134138249 IC50 = 120 nM T94119 CQ2S4X 134138703 IC50 = 188 nM T94119 CQUY75 134139416 IC50 = 51 nM T94119 CL3Q6G 134140420 IC50 = 130 nM T94119 C0PN3R 134140590 IC50 = 55 nM T94119 CN5VU4 134142014 IC50 = 3.8 nM T94119 CDJ10M 134142931 IC50 = 146 nM T94119 CUE85S 134143151 IC50 = 5600 nM T94119 CN59WG 134143270 IC50 = 1090 nM T94119 CL4E9X 134144824 IC50 = 330 nM T94119 CQ9G7H 134145670 IC50 = 9 nM T94119 C1PVM6 134145863 IC50 = 9100 nM T94119 C6G8EJ 134146051 IC50 = 55000 nM T94119 CIPL93 134147099 IC50 = 110 nM T94119 C8ITR3 134147904 IC50 = 7700 nM T94119 CV2QA7 134148173 IC50 = 1000 nM T94119 CXA3V0 134148445 IC50 = 488 nM T94119 C3FO5C 134149163 IC50 = 740 nM T94119 CY3HC4 134150338 IC50 = 11 nM T94119 CXU92M 134150578 IC50 = 15 nM T94119 CG8LE2 134151667 IC50 < 10000 nM T94119 CK43EY 134152988 IC50 = 22 nM T94119 CL5MR8 134154147 IC50 = 17000 nM T94119 CS2QP7 134154582 IC50 = 16 nM T94119 C2QGB3 134156160 IC50 = 5 nM T94119 CV89ZY 134157127 IC50 = 16 nM T94119 C42RJH 134157534 IC50 = 9 nM T94119 C2SE0Y 134157628 IC50 = 0.2 nM T94119 CDSB36 134248984 IC50 = 0.6166 nM T94119 CKP8O2 134249145 Ki = 7800 nM T94119 CA3U2C 134519452 IC50 = 719 nM T94119 CEO8F9 134519632 IC50 = 106 nM T94119 CKH7O4 134519691 IC50 = 20 nM T94119 CTD03Q 134611885 IC50 = 1.259 nM T94119 CJXA12 134611894 IC50 = 1000 nM T94119 CWZ39C 134823450 IC50 = 1.4 nM T94119 C14AOZ 134823456 IC50 < 1 nM T94119 C54FXD 134957362 IC50 = 158.49 nM T94119 C9FUK2 135151360 IC50 > 30000 nM T94119 CT0GQ6 135197577 IC50 = 0.35 nM T94119 C87VKA 135197594 IC50 = 0.37 nM T94119 CQXS07 135197635 IC50 = 0.23 nM T94119 C7KXF1 135197643 IC50 = 0.18 nM T94119 CY38TL 135391000 IC50 = 2.8 nM T94119 COG86Z 135397763 IC50 = 125.89 nM T94119 CWL67T 135397764 IC50 = 6.31 nM T94119 CX8AI4 135398491 IC50 = 58 nM T94119 CH8TR5 135426721 IC50 = 4000 nM T94119 C7SND1 135429301 IC50 < 100 nM T94119 C6AZ2R 135435018 IC50 = 25118.86 nM T94119 C3QJ8W 135566371 IC50 = 9 nM T94119 C24ZGX 135566644 IC50 = 1395 nM T94119 C2QDV5 135566741 IC50 = 118 nM T94119 C2UN0D 135742360 IC50 = 6400 nM T94119 CU29YK 135750268 IC50 = 84 nM T94119 C02PHA 135927892 IC50 = 6309.57 nM T94119 CS8T3D 135927897 IC50 = 501.19 nM T94119 C12UDA 135947972 IC50 = 161 nM T94119 CN42ZS 135947973 IC50 = 250 nM T94119 CF8AO3 135947974 IC50 = 90 nM T94119 CW08GJ 135947976 IC50 = 66 nM T94119 C8O9HG 135947977 IC50 = 100000 nM T94119 CJN7E2 135947978 IC50 = 61 nM T94119 CFKH34 135947979 IC50 = 59 nM T94119 C0ZH9X 135981194 IC50 = 25560 nM T94119 C4G2HP 135995897 IC50 = 1680 nM T94119 CNF15Q 135995898 IC50 = 320 nM T94119 C98HZG 135995899 IC50 = 1020 nM T94119 CIQ82W 135995900 IC50 = 880 nM T94119 CD57NX 136027097 Ki = 2.85 nM T94119 CP1US5 136041737 IC50 = 164 nM T94119 CXH63V 136041747 IC50 = 219 nM T94119 C6B5TC 136041748 IC50 = 779 nM T94119 CU6XG1 136041749 IC50 = 442 nM T94119 C0U5DB 136041750 IC50 = 397 nM T94119 C48KAQ 136041752 IC50 = 9040 nM T94119 C74PRL 136041753 IC50 = 854 nM T94119 CT4FJ1 136041757 IC50 = 28 nM T94119 CCS2G6 136041761 IC50 = 1137 nM T94119 CEZP21 136041762 IC50 = 855 nM T94119 CJ58TD 136041764 IC50 = 2555 nM T94119 CX67QW 136041765 IC50 = 36 nM T94119 CK0H2Q 136041766 IC50 = 84 nM T94119 CQP7B6 136041767 IC50 = 3360 nM T94119 CM65BS 136041773 IC50 = 225 nM T94119 C6P7JB 136041775 IC50 = 247 nM T94119 C5CJF7 136041776 IC50 = 36 nM T94119 C3XIZ8 136041777 IC50 = 270 nM T94119 C32LKO 136041785 IC50 = 2210 nM T94119 C90ARP 136041787 IC50 = 2850 nM T94119 CZ3BN1 136041792 IC50 = 122 nM T94119 CG19DI 136041799 IC50 = 21 nM T94119 CXJA29 136041804 IC50 = 87 nM T94119 CHT31V 136041805 IC50 = 17 nM T94119 CO8C4J 136041817 IC50 = 6 nM T94119 C4QU6G 136041827 IC50 = 4135 nM T94119 CNE10X 136041834 IC50 = 648 nM T94119 CS3AE1 136041847 IC50 = 86 nM T94119 CZC47Y 136041848 IC50 = 278 nM T94119 CA91JG 136069599 IC50 = 18 nM T94119 CGAB91 136069600 IC50 = 34 nM T94119 C3ZAW2 136069605 IC50 = 98 nM T94119 C8JXL5 136069609 IC50 = 22 nM T94119 C9I0EQ 136069610 IC50 = 106 nM T94119 C25EYJ 136069611 IC50 = 7 nM T94119 C2S5QF 136069615 IC50 = 2 nM T94119 CC4UM3 136176116 IC50 = 180 nM T94119 CJRK81 136176117 IC50 = 274 nM T94119 C63IOS 136176118 IC50 = 181 nM T94119 C3KW7H 136176119 IC50 = 6748 nM T94119 C69AKQ 136176120 IC50 = 3406 nM T94119 CF17KO 136176121 IC50 = 8450 nM T94119 CU3TE0 136176122 IC50 = 2755 nM T94119 C3X5KE 136176124 IC50 = 2385 nM T94119 CA8C5E 136176125 IC50 = 2271 nM T94119 C5OMG2 136176126 IC50 = 373 nM T94119 CP2YM7 136176127 IC50 = 1181 nM T94119 C8XIJ0 136176128 IC50 = 398 nM T94119 CUY8N4 136176129 IC50 = 2170 nM T94119 C3J4ME 136176130 IC50 = 335 nM T94119 CR1NZ2 136176131 IC50 = 995 nM T94119 C4WG2F 136176132 IC50 = 151 nM T94119 CJ8EC5 136176139 IC50 = 1060 nM T94119 CQ84IZ 136180335 Ki > 4000 nM T94119 C1LK9U 136183381 IC50 = 55 nM T94119 C27TKQ 136196449 IC50 = 22 nM T94119 CK9S4X 136229137 IC50 = 140 nM T94119 C7S1YJ 136230225 IC50 = 2450 nM T94119 C3Q6ED 136230226 IC50 = 1108 nM T94119 CKPF02 136230227 IC50 = 4270 nM T94119 CZY9O0 136230228 IC50 = 2783 nM T94119 CRET01 136230229 IC50 = 611 nM T94119 CX1KI8 136230230 IC50 = 189 nM T94119 C3Z5MH 136230231 IC50 = 135 nM T94119 CUE6N8 136230232 IC50 = 63 nM T94119 C8Q1AP 136230233 IC50 = 137 nM T94119 C70RXE 136230234 IC50 = 148 nM T94119 C4W0KN 136230235 IC50 = 297 nM T94119 CMZN01 136230236 IC50 = 4647 nM T94119 CCU0H5 136241428 IC50 = 24 nM T94119 C4QMY7 136244246 IC50 = 11530 nM T94119 CF3DK1 136245085 IC50 = 24030 nM T94119 CEU87Z 136245089 IC50 = 580 nM T94119 CI6HG4 136249373 IC50 = 449 nM T94119 CL4MO3 136249382 IC50 = 278 nM T94119 C04LZP 136254186 IC50 = 29730 nM T94119 C8PT7R 136254187 IC50 > 100000 nM T94119 CCJV79 136254188 IC50 > 100000 nM T94119 C5QE8W 136254189 IC50 = 18970 nM T94119 C0GZV9 136254283 IC50 = 2870 nM T94119 CMWA86 136264282 IC50 = 36 nM T94119 CSD78N 136264452 IC50 = 1530 nM T94119 C1HI5T 136264454 IC50 = 21 nM T94119 CV3UE9 137333450 EC50 = 4.3 nM T94119 CH8WU5 137348751 IC50 = 0.7943 nM T94119 CH24ZD 137631369 IC50 = 2.4 nM T94119 CP34TI 137631388 IC50 = 7.4 nM T94119 CF0PQ2 137632018 IC50 = 1.585 nM T94119 C3XH0L 137632431 IC50 > 300 nM T94119 CF4JC7 137632807 IC50 = 110 nM T94119 CIX4S7 137633081 IC50 = 0.7943 nM T94119 CPG41O 137633365 IC50 = 120 nM T94119 C3ST1Q 137633684 IC50 = 1.259 nM T94119 CQ48RD 137633874 IC50 < 0.3 nM T94119 CA4MB6 137633919 IC50 = 10.7 nM T94119 CZ8Q6V 137634548 IC50 = 7200 nM T94119 CGO01Z 137634959 IC50 = 141 nM T94119 C9GXM1 137635017 IC50 = 1 nM T94119 C06BDR 137635072 IC50 = 11 nM T94119 CY86AJ 137635564 IC50 = 19.95 nM T94119 C5GHK7 137635800 IC50 = 16.8 nM T94119 CYK6C4 137635941 IC50 = 1 nM T94119 CMN6T7 137636115 IC50 = 6.73 nM T94119 CZ74XF 137636132 IC50 = 1.259 nM T94119 CPJ43Y 137636841 IC50 = 9.8 nM T94119 C1PVW6 137637361 IC50 > 300 nM T94119 CXPI97 137637422 IC50 = 6.31 nM T94119 CP2J4D 137638455 IC50 = 97.7 nM T94119 C83VBZ 137639018 IC50 = 6.6 nM T94119 CMZV19 137639099 IC50 = 1 nM T94119 CJ3LX4 137639119 IC50 = 9.4 nM T94119 CS78JW 137639139 IC50 = 16 nM T94119 CM4HB3 137639229 IC50 = 4.3 nM T94119 C8A2SJ 137639272 IC50 > 300 nM T94119 C4U8LN 137639297 IC50 = 9.6 nM T94119 C1UZ4S 137639310 IC50 = 44 nM T94119 CBK6W4 137639515 IC50 = 10100 nM T94119 CY52QL 137639725 IC50 = 2700 nM T94119 C4TSZ8 137639858 IC50 = 3.981 nM T94119 CKI6W2 137640126 IC50 = 240 nM T94119 C9EN8L 137640131 IC50 = 4.2 nM T94119 C7HA4V 137640279 IC50 = 10 nM T94119 CA0QO6 137640453 IC50 = 3.82 nM T94119 C37IUP 137640698 IC50 = 2700 nM T94119 C67NLM 137640896 IC50 = 12.59 nM T94119 CPW4L0 137641184 IC50 = 440 nM T94119 C2M1DL 137641375 IC50 = 3070 nM T94119 CQ8X0E 137641383 IC50 = 34 nM T94119 C0I6RQ 137641405 IC50 = 10 nM T94119 C8N1XG 137641715 IC50 = 135 nM T94119 CN3F5A 137641753 IC50 = 1.995 nM T94119 CLA7J8 137642251 IC50 = 12.2 nM T94119 C5X3TH 137642662 IC50 = 29 nM T94119 C8M9TX 137642801 IC50 = 29 nM T94119 CL4Q9G 137643238 IC50 = 2.512 nM T94119 CKU69P 137643285 IC50 = 50.12 nM T94119 CP3JK1 137643598 IC50 = 19.95 nM T94119 CE79MN 137643690 IC50 = 112 nM T94119 CV97OC 137644428 IC50 = 100 nM T94119 CAPQ93 137644458 IC50 = 20 nM T94119 CQSG70 137644855 IC50 = 107 nM T94119 C80WHF 137645205 IC50 = 620 nM T94119 CMYG31 137645705 IC50 = 43 nM T94119 CX8R1L 137645813 IC50 = 188 nM T94119 CID85J 137646014 IC50 = 70 nM T94119 C6SW7U 137646075 IC50 = 1.995 nM T94119 C5ERV3 137646413 IC50 = 27 nM T94119 CZC27Y 137646667 IC50 = 2.512 nM T94119 C3BM5S 137646790 IC50 = 1.4 nM T94119 CA4V8H 137646998 IC50 = 2.512 nM T94119 C9U0CF 137647045 IC50 = 5800 nM T94119 C5HIM9 137647114 IC50 = 2.512 nM T94119 CPMG65 137647250 IC50 = 0.87 nM T94119 C9K7OS 137647525 IC50 = 150 nM T94119 C3TXN9 137647591 IC50 = 13.8 nM T94119 CPX42N 137647765 IC50 = 15 nM T94119 C1FV9C 137647875 IC50 = 0.8 nM T94119 CI3UE7 137647995 IC50 = 41.5 nM T94119 CS39XP 137648085 IC50 = 1.585 nM T94119 C4Z0NQ 137648826 IC50 = 0.7943 nM T94119 CE54DO 137648917 IC50 = 5.012 nM T94119 CSML14 137649696 IC50 = 3 nM T94119 C9FAK1 137650131 IC50 = 0.3 nM T94119 C1R2BI 137650375 IC50 > 300 nM T94119 CUC02Z 137650404 IC50 = 5680 nM T94119 CHT1R8 137650579 IC50 = 2.512 nM T94119 CM8HZ3 137650719 IC50 = 1 nM T94119 CQ3KH9 137650741 IC50 = 4000 nM T94119 C5WR6T 137651215 IC50 = 0.9 nM T94119 CVEL76 137651324 IC50 = 2800 nM T94119 CS2RU9 137652004 IC50 = 170 nM T94119 C7PL6S 137652682 IC50 = 1.3 nM T94119 C9QA0W 137652944 IC50 = 12.59 nM T94119 C38FXZ 137653443 IC50 < 0.2 nM T94119 C1K6TD 137653515 IC50 = 11.8 nM T94119 CN78RE 137653565 IC50 = 0.7943 nM T94119 CTKQ38 137653713 IC50 = 39.81 nM T94119 CI26PN 137653800 IC50 = 9200 nM T94119 C13JPX 137654370 IC50 < 0.3 nM T94119 C9O7ZD 137654904 IC50 > 300 nM T94119 CD19ZS 137654937 IC50 = 4.9 nM T94119 C4N5LS 137655123 IC50 = 7.943 nM T94119 C29HVQ 137655302 IC50 = 4.5 nM T94119 CJNL46 137655684 IC50 = 1.4 nM T94119 CP4S1L 137655824 IC50 = 11.5 nM T94119 CHV26G 137655828 IC50 = 1.1 nM T94119 CC5NK4 137655965 IC50 = 2.512 nM T94119 C5T9JU 137656472 IC50 = 20 nM T94119 CLC7N4 137656507 IC50 = 1.585 nM T94119 CE9H8D 137657006 IC50 = 3.981 nM T94119 C1YN2Q 137657270 IC50 = 78.1 nM T94119 C1K4TB 137657388 IC50 = 14700 nM T94119 C2JX1W 137657572 IC50 = 3.162 nM T94119 C2D0TG 137657839 IC50 = 19.6 nM T94119 C41OPW 137658031 IC50 = 19.95 nM T94119 C6IR2E 137658119 IC50 = 2700 nM T94119 CU15TO 137658167 IC50 = 107 nM T94119 CCX72Y 137658365 IC50 = 60.2 nM T94119 C6BF8E 137658458 IC50 = 23 nM T94119 CI10RD 137658475 IC50 = 30 nM T94119 C90PIR 137658553 IC50 = 2900 nM T94119 CSB1U0 137658705 IC50 = 0.4 nM T94119 C03QAR 137659338 IC50 = 96.8 nM T94119 C5T8OX 137659620 IC50 > 300 nM T94119 C3CF4O 137659746 IC50 = 6.31 nM T94119 C49BSM 137659860 IC50 = 67.1 nM T94119 C1F6QN 137660818 IC50 = 1.259 nM T94119 C34WTV 137660874 IC50 = 5 nM T94119 CP5K4E 137660883 IC50 = 7.1 nM T94119 C1OLQ3 137660961 IC50 = 3.162 nM T94119 CM6FS2 137661095 IC50 = 1.585 nM T94119 C8R3JK 137661301 IC50 = 0.631 nM T94119 C6KR2A 137661344 IC50 = 80.2 nM T94119 C9HPG8 137661516 IC50 = 120 nM T94119 CKDZ26 138504497 IC50 = 800 nM T94119 C2T8OY 138857923 IC50 = 10 nM T94119 CPQ87J 139410792 IC50 < 20 nM T94119 C7ZAQ1 141406387 IC50 = 38160 nM T94119 C7NUI8 141406388 IC50 = 67810 nM T94119 CQYI18 141406390 IC50 = 11160 nM T94119 CUA1D0 141406392 IC50 = 56190 nM T94119 CP0R6Y 141406393 IC50 = 3910 nM T94119 C1EVQ0 141406394 IC50 = 23680 nM T94119 C2QP0F 141406396 IC50 = 44740 nM T94119 CY2M0B 141406399 IC50 = 8140 nM T94119 CC3OU2 141406400 IC50 = 47920 nM T94119 CKV13Y 141406404 IC50 = 28610 nM T94119 C3Q1VL 141419885 IC50 = 2.7 nM T94119 C3FPW6 141419887 IC50 = 7.8 nM T94119 C3EJX8 141419888 IC50 = 3.1 nM T94119 CKX4P3 141446054 IC50 = 7943.28 nM T94119 CV54CS 141471198 IC50 = 4.2 nM T94119 C25HYI 141471200 IC50 = 2.7 nM T94119 CZS03J 141509623 IC50 = 275 nM T94119 CFD94N 141754136 IC50 = 0.7 nM T94119 CX0E9B 142505968 IC50 = 68 nM T94119 C9G5ZW 142505990 IC50 = 5 nM T94119 CBJC50 142505992 IC50 = 49 nM T94119 CJ5GT3 142506013 IC50 = 0.7 nM T94119 C7N8LV 142506025 IC50 = 46 nM T94119 CKBF56 142506033 IC50 < 5 nM T94119 CQ34YR 142506035 IC50 = 81 nM T94119 CU03GW 142506036 IC50 = 4 nM T94119 C74MXW 142506065 IC50 = 0.7 nM T94119 C1PNM8 142506077 IC50 = 663 nM T94119 CX6BQ7 142506102 IC50 = 0.2 nM T94119 CY3BM0 142506119 IC50 = 96 nM T94119 CFJ6X3 142506136 IC50 = 133 nM T94119 CC6MD0 142506155 IC50 = 5 nM T94119 C05QOM 142506157 IC50 = 41 nM T94119 CLND62 142506170 IC50 = 520 nM T94119 CGNQ74 142506189 IC50 = 47 nM T94119 CT3U9R 142506192 IC50 = 0.2 nM T94119 CP71ZJ 142506208 IC50 = 189 nM T94119 C1T3IQ 142506210 IC50 = 0.2 nM T94119 CEGV67 142506220 IC50 = 0.6 nM T94119 CP5HF8 142506225 IC50 = 49 nM T94119 C1U3CA 142506238 IC50 = 32 nM T94119 C7QMG9 145108300 IC50 = 6.8 nM T94119 CGF4I3 145946093 IC50 = 5.012 nM T94119 CJ70MV 145946114 IC50 = 1 nM T94119 CI40JE 145951013 IC50 = 25.6 nM T94119 C6YT8E 145951131 IC50 = 5390 nM T94119 CFW62M 145951569 IC50 = 5.3 nM T94119 CHA84K 145951830 IC50 = 420.4 nM T94119 CT4I9A 145952160 IC50 = 53.9 nM T94119 C91GVH 145952598 IC50 = 1 nM T94119 C1W0GJ 145952796 IC50 = 19952.62 nM T94119 CY18SN 145953214 Ki = 20 nM T94119 CVMF13 145953272 IC50 = 2134 nM T94119 CYL5T1 145953372 IC50 <= 10000 nM T94119 CP14AV 145953653 IC50 = 751 nM T94119 CY8D5Q 145953886 IC50 = 10 nM T94119 C3ZUW8 145954195 IC50 = 156.5 nM T94119 C1NJB7 145955070 IC50 = 3 nM T94119 CRHE01 145955133 IC50 <= 10000 nM T94119 C7MP9Z 145955279 IC50 = 1.4 nM T94119 C7K8VT 145955565 IC50 = 6.2 nM T94119 CPU4X2 145955670 IC50 = 100.4 nM T94119 C3ST5Y 145955693 IC50 = 2 nM T94119 C1VH5X 145955836 IC50 = 20.5 nM T94119 CGHE02 145956080 Ki = 12 nM T94119 C7K2YF 145956631 IC50 <= 10000 nM T94119 CQW74M 145956683 IC50 = 3.3 nM T94119 CJ1F6A 145956725 IC50 = 135.2 nM T94119 C12IFO 145956886 IC50 = 8.6 nM T94119 C9O2PL 145958063 IC50 = 3.2 nM T94119 CQH01X 145958257 IC50 <= 10000 nM T94119 C3DGU7 145958571 IC50 = 1.3 nM T94119 C9NS6T 145958690 IC50 = 11.5 nM T94119 C7ZO9V 145959196 IC50 = 109.4 nM T94119 CSC81H 145959429 IC50 = 2.1 nM T94119 C0S1YM 145959980 IC50 = 21 nM T94119 CT3I2R 145960112 IC50 = 100 nM T94119 C8MJ9X 145960272 IC50 = 15 nM T94119 CF36RA 145961004 IC50 = 2 nM T94119 CHF56O 145961403 IC50 = 374 nM T94119 C2GT9Y 145961404 IC50 = 65 nM T94119 CAI0D6 145963117 IC50 = 87.8 nM T94119 CG6FW9 145967821 IC50 = 4.4 nM T94119 C9NH1Z 145967866 IC50 = 18.7 nM T94119 CCPB17 145967913 IC50 = 2.9 nM T94119 CB43FK 145968534 IC50 = 3 nM T94119 CGL03I 145969468 IC50 = 4.6 nM T94119 C2MST5 145969505 IC50 = 13.5 nM T94119 C97IKW 145969580 IC50 = 4.5 nM T94119 CK82QG 145969816 IC50 = 4364 nM T94119 C71YAK 145970017 IC50 = 10000 nM T94119 CKVI18 145970638 IC50 = 5.5 nM T94119 CTQ50N 145970860 IC50 = 5.5 nM T94119 CZ98FH 145971490 IC50 = 291.5 nM T94119 CTB97Z 145971948 IC50 = 11.5 nM T94119 CGQJ04 145972017 IC50 = 375.9 nM T94119 CA7X9N 145973949 IC50 = 307 nM T94119 CZ9G6E 145974533 IC50 = 12.3 nM T94119 C3LR4O 145976442 IC50 = 8672 nM T94119 CPZS56 145982349 EC50 = 19100 nM T94119 C3UWH8 145982505 IC50 = 84 nM T94119 C9UB4R 145982673 IC50 = 81 nM T94119 COI5P8 145982999 IC50 = 106 nM T94119 CH90CT 145983168 IC50 = 425.2 nM T94119 C1GLK2 145983578 IC50 = 86 nM T94119 CJU02I 145983624 IC50 = 8.4 nM T94119 CVS2U0 145983808 IC50 = 8.6 nM T94119 C6QL4V 145983880 IC50 = 16 nM T94119 CL6HZ9 145983897 IC50 = 227 nM T94119 CL0ZO7 145984847 IC50 = 26 nM T94119 CBTH68 145985019 IC50 = 41 nM T94119 C1HO7R 145986167 IC50 = 31 nM T94119 CP0IX3 145986185 IC50 = 416 nM T94119 CF8MR5 145986347 IC50 = 5000 nM T94119 C06ELG 145987952 IC50 = 3.4 nM T94119 CF82DR 145988183 IC50 = 8.1 nM T94119 CN0DH1 145989043 IC50 = 5.2 nM T94119 C6XMQ8 145989163 EC50 = 15670 nM T94119 CP8TH4 145989722 IC50 = 17 nM T94119 C8X2IT 145996536 IC50 = 1700 nM T94119 C6RPG0 146014481 IC50 = 7.413 nM T94119 C59KOM 146585662 IC50 = 7 nM T94119 CFQO97 146585699 IC50 = 60 nM T94119 C0GMR1 146585718 IC50 = 26 nM T94119 CI85VS 146731761 IC50 = 120 nM T94119 C4MC0S 149169124 IC50 = 4620 nM T94119 CVW62P 149242889 IC50 = 23680 nM T94119 CN87RZ 149370890 IC50 = 1420 nM T94119 CK4FJ1 149556361 IC50 = 7510 nM T94119 C8UQL4 153940691 IC50 = 750 nM T94119 CMZ68Q 153940692 IC50 = 420 nM T94119 C5X7JK 154734328 IC50 = 10 nM T94119 C69VNW 155510695 IC50 = 1584.89 nM T94119 C8Q9UG 155510876 IC50 = 390 nM T94119 CDT8F2 155510913 IC50 = 251.19 nM T94119 CQP9K0 155510991 IC50 = 970 nM T94119 CT6WX1 155511199 IC50 = 32 nM T94119 C9ZL7Y 155511258 IC50 = 11 nM T94119 CH12LB 155511310 IC50 = 374 nM T94119 C1OR2T 155511706 IC50 = 1000 nM T94119 C6PZ9F 155511758 IC50 = 540 nM T94119 C6WIC9 155511977 IC50 = 316.23 nM T94119 CPH8N1 155512095 IC50 = 3.162 nM T94119 CVX7Y0 155512208 IC50 = 33 nM T94119 CZJ9D6 155512258 IC50 = 24 nM T94119 CG9I4X 155512515 IC50 = 230 nM T94119 CR1Z8A 155512529 IC50 = 38 nM T94119 CD36LK 155512654 IC50 = 42 nM T94119 CQZY50 155512775 IC50 = 6.31 nM T94119 C5V2GO 155512947 IC50 = 398.11 nM T94119 C5GWL0 155513019 IC50 = 0.99 nM T94119 C1DIT4 155513047 IC50 = 50.12 nM T94119 C8PG6Z 155513084 IC50 = 158.49 nM T94119 C5M6NS 155513226 IC50 = 9.5 nM T94119 CZG6K5 155513391 IC50 = 60 nM T94119 C45SYX 155513615 IC50 = 2.2 nM T94119 C4UZI2 155514046 IC50 = 31622.78 nM T94119 C96VIE 155514302 IC50 = 11 nM T94119 CB81DS 155514349 IC50 = 6.2 nM T94119 C34VCY 155514382 IC50 = 8.4 nM T94119 CQ1X6F 155514587 IC50 = 42 nM T94119 CBH57O 155514764 IC50 = 125.89 nM T94119 C5C9EG 155515047 IC50 = 79.43 nM T94119 CEFS61 155515135 IC50 = 4720 nM T94119 CR1XO3 155515353 IC50 = 1258.93 nM T94119 C0AXF7 155515394 IC50 = 199.53 nM T94119 CXTC52 155515425 IC50 = 12589.25 nM T94119 CN1T7S 155515661 IC50 = 163 nM T94119 C7Q3FR 155515734 IC50 = 79.43 nM T94119 CL45GQ 155516260 IC50 = 1000 nM T94119 C5IR0K 155516391 IC50 = 2.4 nM T94119 C30ZFN 155516445 IC50 = 316.23 nM T94119 CJDG04 155516604 IC50 = 15.85 nM T94119 CRPB20 155516993 IC50 = 689 nM T94119 C42JXQ 155517064 IC50 = 199.53 nM T94119 CYO19V 155517071 IC50 = 158.49 nM T94119 CVY7O4 155517153 IC50 = 1.8 nM T94119 CYWX76 155517213 IC50 = 50.12 nM T94119 COE6G3 155517381 IC50 = 38 nM T94119 C0D3NR 155517424 IC50 = 25118.86 nM T94119 CT53XD 155517442 IC50 = 1584.89 nM T94119 C4G8YN 155517534 IC50 = 57 nM T94119 CS2JT9 155518175 IC50 = 1995.26 nM T94119 CW9GU4 155518188 IC50 = 1.7 nM T94119 CW7OM6 155518918 IC50 = 44 nM T94119 CC51GM 155519635 IC50 = 79.43 nM T94119 CMB6L0 155519660 IC50 = 343 nM T94119 CHFJ25 155519726 IC50 = 3.162 nM T94119 CZ78HW 155519830 IC50 = 79.43 nM T94119 CQEK39 155520373 IC50 = 6.8 nM T94119 C62TIK 155520386 IC50 = 29 nM T94119 C3D7FJ 155520444 IC50 = 3.162 nM T94119 C46YUA 155521057 IC50 = 87 nM T94119 C5D6YX 155521099 IC50 = 8100 nM T94119 C9N0YC 155521102 IC50 = 1.9 nM T94119 CEA3M1 155521494 IC50 = 25.12 nM T94119 CQD23C 155521715 IC50 = 2 nM T94119 CYI0T6 155521865 IC50 = 94 nM T94119 CBSR95 155522042 IC50 = 9490 nM T94119 CZO7Q8 155522149 IC50 = 44 nM T94119 CY0HL3 155522306 IC50 = 37 nM T94119 CCGW06 155523124 IC50 = 125.89 nM T94119 CNB70P 155523246 IC50 = 398.11 nM T94119 C4TLQ7 155523447 IC50 = 7 nM T94119 CO4S8X 155523501 IC50 > 10000 nM T94119 CZG27I 155523570 IC50 = 421 nM T94119 C37RVF 155523599 IC50 = 64 nM T94119 C4H2AB 155524238 IC50 = 12.59 nM T94119 CP18VT 155524467 IC50 = 12.59 nM T94119 C2PJ0X 155524583 IC50 = 89 nM T94119 C9VN1E 155524769 IC50 = 530 nM T94119 CUP7L2 155524901 IC50 = 100 nM T94119 C2BL5I 155525312 IC50 = 5.012 nM T94119 CE2OM4 155525333 IC50 = 3981.07 nM T94119 C10RZQ 155525477 IC50 = 19.95 nM T94119 CF76OV 155525717 IC50 = 3.9 nM T94119 CV21MY 155525971 IC50 = 39 nM T94119 C0UA4D 155525996 IC50 = 39.81 nM T94119 C0AR4W 155526097 IC50 = 5011.87 nM T94119 CD53VX 155526104 IC50 = 6.8 nM T94119 CNHS85 155526193 IC50 = 7943.28 nM T94119 C3EAR8 155526323 IC50 = 31.62 nM T94119 CFSJ40 155526749 IC50 = 0.93 nM T94119 CFHZ79 155527103 IC50 = 45 nM T94119 CK73QV 155527272 IC50 = 4.7 nM T94119 COU62P 155527495 IC50 = 31 nM T94119 C82NUW 155527501 IC50 = 38 nM T94119 CK07GS 155527559 IC50 = 38 nM T94119 CX12MK 155527651 IC50 = 4 nM T94119 CD89EL 155528247 IC50 = 3 nM T94119 CB9IO8 155528449 IC50 = 20 nM T94119 C8Z3TK 155528581 IC50 = 63.1 nM T94119 C0B2NV 155528644 IC50 = 3.2 nM T94119 COY5G1 155528831 IC50 = 58 nM T94119 CF1MS3 155528972 IC50 = 28.3 nM T94119 C3VAI9 155528997 IC50 = 251.19 nM T94119 C2FE1S 155529479 IC50 = 7.943 nM T94119 CB90AR 155529643 IC50 = 125.89 nM T94119 CFV1S0 155529706 IC50 = 40 nM T94119 C3XLY2 155529766 IC50 = 153 nM T94119 C14QOF 155530163 IC50 = 25.12 nM T94119 C4I5UP 155530224 IC50 = 158.49 nM T94119 CZL26X 155530501 IC50 = 18 nM T94119 CW24QE 155531054 IC50 = 576 nM T94119 CX6N3Y 155531155 IC50 = 79.43 nM T94119 C9AXO7 155531257 IC50 = 79.43 nM T94119 CGAI60 155531409 IC50 = 3.981 nM T94119 CDI4V8 155531526 IC50 = 34 nM T94119 CE6QP1 155532037 IC50 = 10 nM T94119 CJH9U4 155532237 IC50 = 1258.93 nM T94119 C6W0JX 155532471 IC50 = 501.19 nM T94119 CIM18N 155532540 IC50 = 28 nM T94119 CKMD29 155532546 IC50 = 125.89 nM T94119 CNMC95 155532794 IC50 = 11.1 nM T94119 C3XFB8 155532820 IC50 = 12.59 nM T94119 C0GR1J 155533050 IC50 = 0.7 nM T94119 CQS8P1 155533070 IC50 = 125.89 nM T94119 C0SZR9 155533335 IC50 = 150 nM T94119 CAT9V1 155533370 IC50 = 3 nM T94119 C67ERP 155533384 IC50 = 100 nM T94119 CL8OM7 155533564 IC50 = 4 nM T94119 CBM24U 155533579 IC50 = 125.89 nM T94119 CR5H8B 155533591 IC50 = 79.43 nM T94119 CA7T0Y 155533911 IC50 > 10000 nM T94119 C8XQ4W 155534168 IC50 = 0.2 nM T94119 CN1ST4 155534269 IC50 = 39.81 nM T94119 CDQY81 155534313 IC50 = 4 nM T94119 CBEG39 155534594 IC50 = 199.53 nM T94119 C3MT9C 155534643 IC50 = 150 nM T94119 C59SQY 155534735 IC50 = 27 nM T94119 CCXP81 155535236 IC50 = 180 nM T94119 CG1JR7 155535513 IC50 = 501.19 nM T94119 CN6KJ5 155535520 IC50 = 12.59 nM T94119 C8N6MT 155535532 IC50 = 10000 nM T94119 C5F2TY 155535537 IC50 = 19.95 nM T94119 CKB2U4 155535691 IC50 = 39.81 nM T94119 CY7X3M 155535740 IC50 = 12.59 nM T94119 CUWE49 155535963 IC50 = 630.96 nM T94119 C70UDF 155536179 IC50 = 125.89 nM T94119 CEJ6L1 155536226 IC50 = 3.7 nM T94119 CNB24M 155536473 IC50 = 25.12 nM T94119 CI6L8Q 155536677 IC50 = 26 nM T94119 CDF3T9 155536730 IC50 = 22 nM T94119 C2CG1A 155537016 IC50 = 251.19 nM T94119 CSO87C 155537103 IC50 = 12 nM T94119 CS24EV 155537776 IC50 = 110 nM T94119 C34SNT 155537955 IC50 = 58 nM T94119 C8AJ6C 155538256 IC50 = 1.3 nM T94119 CQ1E6H 155538266 IC50 = 15.85 nM T94119 CZ19AN 155538609 IC50 = 171 nM T94119 CHR8M1 155538990 IC50 = 9760 nM T94119 CZ9B1L 155539017 IC50 = 2.8 nM T94119 CC1BG2 155539321 IC50 = 25 nM T94119 CF20PS 155539394 IC50 = 100 nM T94119 CUC3F8 155539997 IC50 = 3.2 nM T94119 CL8NI2 155540037 IC50 = 23 nM T94119 C8LKW4 155540264 IC50 = 25.12 nM T94119 CKX3G2 155540908 IC50 = 7.2 nM T94119 C6I5DK 155541290 IC50 = 501.19 nM T94119 CI8XL2 155541479 IC50 = 9.6 nM T94119 CECX47 155541544 IC50 = 1.585 nM T94119 C7A3SN 155541583 IC50 = 49 nM T94119 C2D4ZP 155541609 IC50 = 7943.28 nM T94119 C4FC0V 155541900 IC50 = 251.19 nM T94119 C57MVO 155542051 IC50 = 5011.87 nM T94119 CASE16 155542363 IC50 = 794.33 nM T94119 C8AXF9 155542633 IC50 = 398.11 nM T94119 C8OC2P 155542800 IC50 = 320 nM T94119 C42BIZ 155542813 IC50 = 1000 nM T94119 CTDQ52 155542836 IC50 = 398.11 nM T94119 CVNR95 155542898 IC50 = 5 nM T94119 C1SY0G 155543154 IC50 = 4.8 nM T94119 C1JRK8 155543277 IC50 = 25118.86 nM T94119 C7IWJ2 155543389 IC50 = 5.012 nM T94119 C1UNH0 155543517 IC50 = 1258.93 nM T94119 CZY0N4 155543588 IC50 = 0.7 nM T94119 C48KXS 155543644 IC50 = 34 nM T94119 CJB8C9 155543659 IC50 = 42 nM T94119 C3CN0A 155543674 IC50 = 7.943 nM T94119 C5MYJ2 155543736 IC50 = 7943.28 nM T94119 CVI3E5 155543933 IC50 = 0.43 nM T94119 C8OSM3 155544223 IC50 = 635 nM T94119 CX1C8I 155544561 IC50 = 8.5 nM T94119 COGF23 155544916 IC50 = 25118.86 nM T94119 C48RPZ 155544941 IC50 = 1000 nM T94119 C98FXC 155544955 IC50 = 50 nM T94119 CW3K4F 155545182 IC50 = 3162.28 nM T94119 C4TYN3 155545535 IC50 = 25118.86 nM T94119 CV8G5R 155545946 IC50 = 27 nM T94119 CTSW53 155546042 IC50 = 9.2 nM T94119 C1HKU0 155546330 IC50 = 33 nM T94119 CQ6J7U 155546361 IC50 = 990 nM T94119 CE1A0D 155546906 IC50 = 9.4 nM T94119 C8SQA2 155546999 IC50 = 6.31 nM T94119 C8D4ZH 155547166 IC50 = 316.23 nM T94119 CMY3J7 155547466 IC50 = 231 nM T94119 C2BS7T 155547557 IC50 = 1270 nM T94119 C31GSV 155547741 IC50 = 47 nM T94119 CH1F9K 155547869 IC50 = 5.9 nM T94119 CJAB13 155548110 IC50 = 18.4 nM T94119 CI6KO7 155548518 IC50 = 316.23 nM T94119 CL4F8P 155549003 IC50 = 6.31 nM T94119 CM6S8K 155549098 IC50 = 39.81 nM T94119 CON58B 155549407 IC50 = 27 nM T94119 CFMH09 155549542 IC50 = 179 nM T94119 C4PEJ5 155549895 IC50 = 9310 nM T94119 CFP94J 155550309 IC50 = 199.53 nM T94119 CCX5E2 155550788 IC50 = 180 nM T94119 CZS9Q8 155551405 IC50 = 0.7943 nM T94119 C3QZE7 155551609 IC50 = 20 nM T94119 CFO52S 155551740 IC50 = 252 nM T94119 C5HR2W 155551907 IC50 = 15848.93 nM T94119 CK1JR7 155551961 IC50 = 7.4 nM T94119 CK53PC 155552028 IC50 = 91 nM T94119 CI3Y5U 155552035 IC50 = 22 nM T94119 CUD43T 155552139 IC50 = 14.3 nM T94119 CWJ72T 155552555 IC50 = 220 nM T94119 CXN3Y8 155553327 IC50 = 25.12 nM T94119 CL04BD 155554125 IC50 = 37 nM T94119 CX9C6O 155554180 IC50 = 19.95 nM T94119 CP7L5X 155554538 IC50 = 14 nM T94119 CVH0M1 155554616 IC50 = 4.9 nM T94119 CC13QL 155555170 IC50 = 263 nM T94119 CZX06J 155555458 IC50 = 50.12 nM T94119 C2OGW1 155555483 IC50 = 29 nM T94119 C3UP9A 155555623 IC50 = 3981.07 nM T94119 C3KXR2 155555660 IC50 = 3 nM T94119 C19WIO 155555836 IC50 = 498 nM T94119 CRO5Z3 155556073 IC50 = 7 nM T94119 CH2P4T 155556124 IC50 = 158489.32 nM T94119 CCU8M1 155556480 IC50 = 501.19 nM T94119 CIU29Z 155556576 IC50 = 11 nM T94119 CM3LI6 155556593 IC50 = 143 nM T94119 CZ8CX1 155556887 IC50 = 39.81 nM T94119 CG2FS6 155557123 IC50 = 50.12 nM T94119 CFS63H 155557182 IC50 = 2 nM T94119 CCL48D 155557746 IC50 = 120 nM T94119 C0FE4G 155557988 IC50 = 170 nM T94119 CR8J0E 155558167 IC50 = 79.43 nM T94119 CN96JH 155558197 IC50 = 1000 nM T94119 CSO4M3 155558261 IC50 = 501.19 nM T94119 C52TSP 155558262 IC50 = 144 nM T94119 CB4A1O 155558535 IC50 = 1258.93 nM T94119 C2VGC6 155558733 IC50 = 7.7 nM T94119 CZMI26 155558737 IC50 = 15848.93 nM T94119 CDS2U1 155558931 IC50 = 24 nM T94119 CLS9Y1 155559053 IC50 = 61 nM T94119 CS70ER 155559192 IC50 = 163 nM T94119 C9KX4D 155559215 IC50 = 920 nM T94119 CSF7G4 155559324 IC50 = 2.5 nM T94119 CAQ0X8 155559376 IC50 = 29.4 nM T94119 CMKY39 155559468 IC50 = 15848.93 nM T94119 CAWI85 155559815 IC50 = 8.9 nM T94119 CDI59L 155560058 IC50 = 5.012 nM T94119 CDJ1P2 155560222 IC50 = 3.2 nM T94119 CVG49I 155560688 IC50 = 5450 nM T94119 C5S7AL 155560766 IC50 = 79.43 nM T94119 C2OT6K 155560767 IC50 = 3162.28 nM T94119 CQ7PS9 155560780 IC50 = 7.943 nM T94119 CLO3B1 155561152 IC50 = 20 nM T94119 C8XS0L 155561165 IC50 = 39.81 nM T94119 C72CQG 155561233 IC50 = 15.85 nM T94119 C1INL7 155561328 IC50 = 19.95 nM T94119 C98FHW 155561366 IC50 = 27 nM T94119 CUGI82 155561991 IC50 = 42 nM T94119 C35VQO 155562231 IC50 = 405 nM T94119 CB1T2W 155562315 IC50 > 31622.78 nM T94119 CX6U2T 155562388 IC50 = 79.43 nM T94119 CN4B3D 155562639 IC50 = 25118.86 nM T94119 C5E9TP 155562641 IC50 > 39810.72 nM T94119 CCF4W2 155563986 IC50 = 158.49 nM T94119 CVZ80N 155564202 IC50 = 10 nM T94119 CYD52H 155564883 IC50 = 178 nM T94119 CHK4E8 155565269 IC50 = 63.1 nM T94119 C7PXA0 155565551 IC50 = 6.31 nM T94119 CY4N7O 155565715 IC50 = 3981.07 nM T94119 CVQ6Z4 155565763 IC50 = 100 nM T94119 CA1RX3 155565771 IC50 = 251.19 nM T94119 CQ3AU4 155565828 IC50 = 630.96 nM T94119 CMK4I3 155565845 IC50 = 63.1 nM T94119 C59VPW 155565958 IC50 = 12.59 nM T94119 CAP9F2 155566187 IC50 = 3 nM T94119 CY5SB4 155566208 IC50 = 63.1 nM T94119 CM7E2G 155566279 IC50 = 794.33 nM T94119 C3BNY5 155566309 IC50 = 316.23 nM T94119 C9HR5K 155566863 IC50 = 15848.93 nM T94119 CXE94L 155567270 IC50 = 43 nM T94119 C9KQW3 155567372 IC50 = 14 nM T94119 C98NZE 155567616 IC50 = 19952.62 nM T94119 C1HQ5J 155568324 IC50 = 6.3 nM T94119 CLA46O 155568356 IC50 = 1780 nM T94119 CH2RY0 155568388 IC50 = 150 nM T94119 C7SLR8 155568452 IC50 = 6.31 nM T94119 CT15RN 155568479 IC50 = 1584.89 nM T94119 CM5XO0 155568497 IC50 = 8330 nM T94119 C3VTU8 155568539 IC50 = 1470 nM T94119 CT0BK2 155568581 IC50 = 11.4 nM T94119 C14LVO 155569074 IC50 = 125.89 nM T94119 CFWP17 155569113 IC50 = 22 nM T94119 C1UD4S 155569289 IC50 = 19.95 nM T94119 CXBZ67 155569362 IC50 = 12589.25 nM T94119 CUH38L 155569363 IC50 = 6150 nM T94119 C4H0NE 155569598 IC50 = 100 nM T94119 D00HSJ 10275789 IC50 = 910 nM T94119 D00ZIK 9908783 Ki = 20 nM T94119 D01SSI 24937012 IC50 = 15 nM T94119 D03EHM 24905142 IC50 = 150 nM T94119 D03QQH 16760391 IC50 = 22000 nM T94119 D06DNH 9907093 IC50 = 851 nM T94119 D06HVH 54613583 IC50 = 4700 nM T94119 D06PWI 42623951 IC50 = 7943.28 nM T94119 D07PMP 44187953 IC50 = 14 nM T94119 D08KSQ 11637090 IC50 > 10000 nM T94119 D08NQM 5289247 IC50 = 300 nM T94119 D0H2CM 135565635 IC50 = 100 nM T94119 D0P5TI 58441401 IC50 = 3020 nM T94119 D0R0TW 11964036 IC50 < 0.1 nM T94119 D0S5YV 6852167 IC50 = 77 nM T94119 D0W8XH 9884685 IC50 = 3 nM T94119 D0X1RH 16051023 IC50 = 440 nM T94119 D0Y3OO 11327430 IC50 = 30 nM T20542 D00OWF 5280953 IC50 = 80000 nM T20542 D0NS6I 10037501 IC50 > 10000 nM T20542 D0Q3VZ 135398522 IC50 = 520 nM T20542 CLS29B 46872626 IC50 > 10000 nM T20542 CDK93W 56946894 IC50 = 40 nM T20542 CV63UL 67240318 IC50 > 10000 nM T20542 D0Z5TQ 5924208 IC50 = 4380 nM T77410 CKT02A 5329452 IC50 > 20000 nM T77410 C4RUV5 5329453 IC50 = 2000 nM T77410 CGN7B0 5329457 IC50 = 6500 nM T77410 CPQ31L 25195294 IC50 = 4.9 nM T77410 CU1R9K 44223241 IC50 = 10 nM T77410 C05DWF 44223242 IC50 = 2600 nM T77410 CKH78Y 44223243 IC50 = 150 nM T77410 CZ7N8F 44223244 IC50 > 20000 nM T77410 C2KE9M 44223297 IC50 = 5 nM T77410 CW5MD8 44223299 IC50 = 350 nM T77410 C3ZI8K 44223300 IC50 = 500 nM T77410 CK5T7Z 44223301 IC50 = 20000 nM T77410 C4ZHV5 44223352 IC50 = 500 nM T77410 C61FEN 44223353 IC50 = 250 nM T77410 C8KFN4 44223354 IC50 = 750 nM T77410 CE48DG 44223355 IC50 = 3300 nM T77410 CUG9N6 44223356 IC50 > 20000 nM T77410 CN2QG1 44223357 IC50 = 55 nM T77410 CY8W1U 44577680 IC50 = 450 nM T77410 C8WRS0 44577681 IC50 = 4500 nM T77410 CUO17D 44577719 IC50 > 20000 nM T77410 CMH1K4 44577720 IC50 > 20000 nM T77410 CL28VX 44577751 IC50 > 20000 nM T77410 CCB85P 44577752 IC50 > 20000 nM T77410 C3CD9B 44577754 IC50 > 20000 nM T77410 CR6WO7 44577770 IC50 = 90 nM T77410 CTQI35 44577771 IC50 = 5000 nM T77410 C6MB3W 44577855 IC50 > 20000 nM T77410 D0RF7O 44577753 IC50 = 3000 nM T77410 D0Y0BK 11524144 IC50 = 430 nM T12084 D07DJQ 10219 IC50 = 7800 nM T12084 COC9V5 710899 IC50 = 1500 nM T12084 CAJ75S 885318 IC50 = 1200 nM T12084 CE9LS5 5524574 IC50 = 9200 nM T12084 CH49NS 5524575 IC50 = 1900 nM T12084 CA8V0J 5823053 IC50 = 5700 nM T12084 C18YSR 5934766 IC50 = 640 nM T41955 D04CSZ 1254 EC50 = 3000 nM T41955 D09NAW 60195662 IC50 = 103 nM T41955 D0CO6D 71144018 IC50 = 13 nM T41955 C9V3ZD 16666 EC50 = 10100 nM T41955 C8UPV1 59022 IC50 = 5960 nM T41955 CGH31L 77158 IC50 = 22700 nM T41955 COM60X 77379 IC50 = 21500 nM T41955 CO3T5G 619457 IC50 = 1500 nM T41955 CENX23 2092599 EC50 = 25000 nM T41955 CRHE73 2463055 IC50 = 25118.86 nM T41955 C0Z7RE 2800731 IC50 = 183 nM T41955 C3PA4E 2831519 IC50 = 21600 nM T41955 CS6E7A 6013922 IC50 = 39810.72 nM T41955 C9TN5P 8369884 EC50 = 1985 nM T41955 CP92WJ 9884140 IC50 = 31622.78 nM T41955 CW9VR1 11508468 IC50 = 59000 nM T41955 CH3F1I 11514966 IC50 = 19952.62 nM T41955 CJ0DF2 16035583 IC50 = 1240 nM T41955 CMVH91 16095383 IC50 = 414 nM T41955 C6TIP3 17013221 EC50 = 200 nM T41955 CIS17P 23872112 EC50 > 10000 nM T41955 CA8MH0 25138305 IC50 = 4 nM T41955 CE8CG1 25207770 IC50 = 391 nM T41955 CJ8OR4 25234679 IC50 = 14 nM T41955 C0T2NE 25234681 IC50 = 24 nM T41955 CJG80H 25234753 IC50 = 200 nM T41955 CQR14M 25234755 IC50 = 1262 nM T41955 CJ5Z9G 25234835 IC50 = 463 nM T41955 CL7XI2 25234909 IC50 = 786 nM T41955 C7FBO1 25270198 IC50 = 44000 nM T41955 CRZJ04 32647548 EC50 = 2005 nM T41955 CUN7T0 32920052 EC50 = 0.7 nM T41955 CR7E6B 38347541 EC50 > 10000 nM T41955 C67JKT 42634918 IC50 = 52 nM T41955 C7LC1U 42635101 IC50 = 171 nM T41955 CG97TM 44566598 EC50 > 10000 nM T41955 CGMW85 46867602 IC50 = 12 nM T41955 CXHM52 46894128 IC50 = 18.9 nM T41955 CAC82P 46917506 IC50 = 48.5 nM T41955 CCB95S 46917507 IC50 = 543.7 nM T41955 C9QI7Y 46917509 IC50 = 41.1 nM T41955 CI5B8U 46917583 IC50 = 177.8 nM T41955 C0Y9WA 46917657 IC50 = 457.2 nM T41955 CW36EG 46917659 IC50 = 265.8 nM T41955 C9D4EO 46917737 IC50 = 230.4 nM T41955 CH03TY 46917811 IC50 = 65.9 nM T41955 CP62XY 46917814 IC50 = 44.5 nM T41955 CD19OH 46917815 IC50 = 90.1 nM T41955 CV65QE 46917816 IC50 = 13.3 nM T41955 C4V7FI 46917876 IC50 = 19.5 nM T41955 CFVX07 46917877 IC50 = 22.5 nM T41955 C2TON8 46937329 IC50 = 61 nM T41955 CBV0H3 49765039 IC50 = 15 nM T41955 CB0GS2 49783548 IC50 = 736 nM T41955 C7D1QZ 49783798 IC50 = 104 nM T41955 CBYO37 49783874 IC50 = 70 nM T41955 CH64QM 49783950 IC50 = 57 nM T41955 CA1BM6 49783951 IC50 = 67 nM T41955 CWO85T 49783952 IC50 = 216 nM T41955 CLX8I1 49783955 IC50 = 40 nM T41955 CP0RU7 49783960 IC50 = 122 nM T41955 CB60GV 49784028 IC50 = 0.96 nM T41955 CJ8ED7 49784031 IC50 = 41 nM T41955 CV90SW 49784110 IC50 = 57 nM T41955 CV7H6Q 49784114 IC50 = 27 nM T41955 C8LIN1 49784184 IC50 = 201 nM T41955 C3XQ4D 49784256 IC50 = 14 nM T41955 C9RMY2 49784334 IC50 = 8 nM T41955 CSJ86E 49784335 IC50 = 3.3 nM T41955 C2OC6F 49784336 IC50 = 96 nM T41955 CWB9Q5 49784337 IC50 = 11 nM T41955 CPJ63C 49784413 IC50 = 49 nM T41955 C0ZKY2 49784414 IC50 = 16 nM T41955 C4GTI8 49784659 IC50 = 67 nM T41955 C32MBN 49784743 IC50 = 762 nM T41955 C5S6GX 51136589 EC50 = 3450 nM T41955 C23WVS 53361524 IC50 > 20000 nM T41955 CZT3M9 56949331 IC50 = 15 nM T41955 C18OKB 56952982 IC50 = 46 nM T41955 CA84IS 56952984 IC50 = 18 nM T41955 CH6Y7Q 56964352 IC50 = 36 nM T41955 C81MJQ 57625473 IC50 = 79 nM T41955 CH06EO 59536254 IC50 = 324 nM T41955 COP8X4 59536299 IC50 = 83 nM T41955 C9DAF7 59536331 IC50 = 37 nM T41955 CPE18Y 59536364 IC50 = 14 nM T41955 C7FOW4 59536377 IC50 = 155 nM T41955 C0M3YK 59536383 IC50 = 424 nM T41955 CA01DU 59536398 IC50 = 398 nM T41955 C92SYQ 59536422 IC50 = 1383 nM T41955 CUV34I 59536431 IC50 = 28 nM T41955 CHB0N6 66600758 IC50 = 406 nM T41955 CKO47V 66600938 IC50 = 9859 nM T41955 C1M2QS 66601076 IC50 = 213 nM T41955 CRH62U 66601095 IC50 = 2983 nM T41955 C7P6FA 66601131 IC50 = 8419 nM T41955 C6V1HY 66601188 IC50 = 3720 nM T41955 C7SM5K 66601362 IC50 = 707 nM T41955 CZ82DS 66601372 IC50 = 42 nM T41955 CMZE60 66907318 IC50 = 6.2 nM T41955 CA9K7J 67510371 EC50 = 0.3 nM T41955 CNF2Y3 67510376 EC50 = 1876 nM T41955 COQ6Z0 67510423 EC50 = 3700 nM T41955 CV6P8W 67510427 EC50 = 1235 nM T41955 CVG0E7 67510513 EC50 = 178 nM T41955 C86TRO 67510566 EC50 = 23 nM T41955 CI24RO 67510666 EC50 = 8 nM T41955 CZK74S 67510760 EC50 = 1400 nM T41955 CY46EN 67510848 EC50 = 8 nM T41955 CHR6C9 67510887 EC50 = 2000 nM T41955 CN9MY7 67510929 EC50 = 97 nM T41955 CM14JK 67510971 EC50 = 88 nM T41955 CI3D8R 67511043 EC50 = 1102 nM T41955 CF2K8B 67511180 EC50 = 120 nM T41955 CF70XQ 67511212 EC50 = 400 nM T41955 C6LRM7 67511214 EC50 = 198 nM T41955 CH9LS8 67511310 EC50 = 192 nM T41955 C3IOU2 67511313 EC50 = 2 nM T41955 CCX9F3 67511470 EC50 = 40 nM T41955 C5GOD1 67511509 EC50 = 10988 nM T41955 CZIU96 67511579 EC50 = 20 nM T41955 CF3G2I 67511619 EC50 = 24 nM T41955 C1R4FW 67511668 EC50 = 2240 nM T41955 CST60F 67511677 EC50 = 120 nM T41955 C6JW5I 67511822 EC50 = 136 nM T41955 CWGZ01 67511908 EC50 = 2 nM T41955 CKCZ82 67512015 EC50 = 93 nM T41955 C1A8DY 67512043 EC50 = 489 nM T41955 CRP94E 67512058 EC50 = 70 nM T41955 CQDM39 67512095 EC50 = 52 nM T41955 CA42KD 67512098 EC50 = 8 nM T41955 CP4C7M 67512148 EC50 = 422 nM T41955 CLA1Y2 67512330 EC50 = 889 nM T41955 C1DW8P 67512362 EC50 = 80 nM T41955 CB98GT 67513371 EC50 = 3062 nM T41955 CW3CH4 67516085 EC50 = 0.3 nM T41955 C8OSA0 67516108 EC50 = 0.2 nM T41955 C12FRY 67516186 EC50 = 0.004 nM T41955 CH52IA 67516291 EC50 = 1.4 nM T41955 CO3PJ6 67516491 EC50 = 1786 nM T41955 C3J7DV 67516631 EC50 = 0.002 nM T41955 CMD94J 67516707 EC50 = 0.8 nM T41955 CS16IK 67516951 EC50 = 0.6 nM T41955 C8YS1K 67517163 EC50 = 0.001 nM T41955 CVM2O5 67517308 EC50 = 422 nM T41955 CSP4Q5 68287829 IC50 = 145 nM T41955 C12ZOH 68287843 IC50 = 234 nM T41955 CO48FM 68287853 IC50 = 94 nM T41955 C2FB8G 68288012 IC50 = 446 nM T41955 C8X1ME 68288092 IC50 = 62 nM T41955 CF2PT6 68288099 IC50 > 5000 nM T41955 C06RFV 68288164 IC50 = 202 nM T41955 CQ5G6W 68288184 IC50 = 3619 nM T41955 CRT18Z 68288237 IC50 = 1159 nM T41955 C1DR6Y 68288249 IC50 = 60 nM T41955 C0X1HO 68288253 IC50 = 328 nM T41955 CO6Z7D 68288263 IC50 = 90 nM T41955 C1JIP7 68288297 IC50 = 123 nM T41955 C9MTL6 68288316 IC50 = 3282 nM T41955 CLF64H 69765682 EC50 = 0.4 nM T41955 CKR75S 71144058 IC50 = 389 nM T41955 CHO4A3 71144083 IC50 = 9 nM T41955 C3CQF5 71144092 IC50 = 5 nM T41955 CK6A9G 71144095 IC50 = 20 nM T41955 CEN1W3 71144099 IC50 = 95 nM T41955 C05SJY 71144244 IC50 = 75 nM T41955 CJO48U 71144284 IC50 = 92 nM T41955 C07VQH 71144348 IC50 = 10 nM T41955 CJMQ52 71144526 IC50 = 75 nM T41955 CS1RN4 71144663 IC50 = 129 nM T41955 C01DIG 71502345 IC50 = 6 nM T41955 C0U2EQ 71502347 IC50 = 27 nM T41955 C8IOE1 71502460 IC50 = 157 nM T41955 C2LPE8 71502545 IC50 = 15 nM T41955 CU4Z3G 71582398 EC50 = 332 nM T41955 C6AS7T 71582399 EC50 = 1150 nM T41955 CP4J0X 71582400 EC50 = 583 nM T41955 C1SKT2 71582401 EC50 = 87 nM T41955 CTR49S 71582490 EC50 = 1130 nM T41955 CCR28P 71582491 EC50 = 82 nM T41955 C3R5HZ 71582492 EC50 = 138 nM T41955 CS5K2W 71582493 EC50 = 329 nM T41955 CK46TH 71582494 EC50 = 66 nM T41955 CNF3V0 71582567 EC50 = 54 nM T41955 CE3QU6 71582570 EC50 = 153 nM T41955 C3QX7D 71801263 IC50 = 2423 nM T41955 C6PJL2 72205120 IC50 = 280.7 nM T41955 CEA51L 72205121 IC50 = 666.9 nM T41955 CQ3DP0 72205303 IC50 = 97.3 nM T41955 CJY68W 72205304 IC50 = 289.6 nM T41955 CTY25S 72205305 IC50 = 113.1 nM T41955 CNXW30 72205306 IC50 = 295.2 nM T41955 CBDN41 72205307 IC50 = 656.9 nM T41955 C26ORT 72205308 IC50 = 182.1 nM T41955 CM4QB6 72205497 IC50 = 111 nM T41955 C6Z5BK 72205498 IC50 = 107.3 nM T41955 C96BEP 72205499 IC50 = 9.5 nM T41955 CXR7L8 72205500 IC50 = 8.9 nM T41955 CO57MJ 72205501 IC50 = 16.6 nM T41955 C74JTD 72205502 IC50 = 94 nM T41955 C8NT4P 72205682 IC50 = 46.3 nM T41955 CDI82J 72205683 IC50 = 60 nM T41955 C3FW8R 72544340 IC50 = 76.2 nM T41955 C8COX1 72545014 IC50 = 3150 nM T41955 C2JA5F 72545015 IC50 = 1230 nM T41955 CC79FP 72545016 IC50 = 1360 nM T41955 CTJV20 72545017 IC50 = 2010 nM T41955 CJEW81 72545018 IC50 = 8780 nM T41955 CCF6U2 72545244 IC50 = 1400 nM T41955 C7QRJ2 72545245 IC50 = 593 nM T41955 CQ5Z8K 72545485 IC50 = 15.1 nM T41955 C6NC4I 72545486 IC50 = 291 nM T41955 C68LSJ 72545487 IC50 = 21.1 nM T41955 C0O7IW 72545488 IC50 = 435 nM T41955 CS1PO8 72545489 IC50 = 29.9 nM T41955 C6T3LD 72545742 IC50 = 85.4 nM T41955 CU0B8W 72545743 IC50 = 96.9 nM T41955 CCH3R7 72545744 IC50 = 19.3 nM T41955 CH2T4S 72545745 IC50 = 254 nM T41955 C9L7NM 72545746 IC50 = 1850 nM T41955 CP0TK2 72545747 IC50 = 493 nM T41955 CZ43QM 72545748 IC50 = 6780 nM T41955 CHV8Y4 86343318 EC50 = 28 nM T41955 CC1VT7 86343319 EC50 = 11 nM T41955 CNJ60K 86687972 IC50 = 18 nM T41955 CKSZ03 86687975 IC50 = 10 nM T41955 CEF81J 87068694 IC50 = 8.9 nM T41955 C8SZU3 89310378 IC50 = 27 nM T41955 CR34PY 89310481 IC50 = 19 nM T41955 C50HKY 89310581 IC50 = 22 nM T41955 C5UY7Z 89310614 IC50 = 35 nM T41955 CX6LP4 89310807 IC50 = 20 nM T41955 CXIT01 89310839 IC50 = 119 nM T41955 CT5O2X 89330114 IC50 = 51 nM T41955 CDQV01 89330124 IC50 = 59 nM T41955 CQV3K7 89609800 EC50 = 86 nM T41955 CYFE92 89642036 IC50 = 8 nM T41955 CN61RW 90645447 IC50 = 9000 nM T41955 CISP03 90645459 IC50 = 17100 nM T41955 CM5FN9 90645460 IC50 = 9200 nM T41955 C31TXQ 90645465 IC50 = 10900 nM T41955 C6OF3B 90645468 IC50 = 4400 nM T41955 C0VW1K 90645470 IC50 = 6400 nM T41955 C6LA4X 90655359 IC50 = 44 nM T41955 CK6Y3I 90655360 IC50 = 154 nM T41955 C1I0VA 90655361 IC50 > 20000 nM T41955 CI2YZ0 90655362 IC50 = 25 nM T41955 CM5C7Q 90655363 IC50 = 53 nM T41955 C9R1ZY 90655364 IC50 = 10 nM T41955 C3OC9H 90655365 IC50 = 48 nM T41955 C6SU4X 90665452 IC50 = 4800 nM T41955 CJCR26 90665456 IC50 = 9580 nM T41955 C5YFP0 91824785 IC50 = 900 nM T41955 C1TL5F 118246688 IC50 = 870 nM T41955 CKPQ15 118246690 IC50 = 5000 nM T41955 C5ACT0 118246707 IC50 = 240 nM T41955 C5IWC0 118246709 IC50 = 400 nM T41955 CZ89PN 118246718 IC50 = 43000 nM T41955 CHL2M3 118246719 IC50 = 19000 nM T41955 CDNC39 118246723 IC50 = 80 nM T41955 C7MR9F 118246755 IC50 = 5600 nM T41955 CE5CU3 118246774 IC50 = 28000 nM T41955 C3Y8SE 118246812 IC50 = 100 nM T41955 C6EW1N 118246884 IC50 = 19000 nM T41955 CR8GY7 118246886 IC50 = 8100 nM T41955 C6PN0X 118246926 IC50 = 11000 nM T41955 CJF20R 118246949 IC50 = 4100 nM T41955 CV5SU0 118246964 IC50 = 2100 nM T41955 CFBX85 118246965 IC50 = 850 nM T41955 CX8CI0 118247015 IC50 = 37000 nM T41955 CR4NT3 118247016 IC50 = 1700 nM T41955 CCF12I 118247022 IC50 = 4700 nM T41955 CML46E 118247023 IC50 = 54000 nM T41955 CP38EG 118247047 IC50 = 390 nM T41955 C9QL7X 118247077 IC50 = 3000 nM T41955 CMS96Z 118247101 IC50 = 180 nM T41955 CI52RV 118719632 IC50 = 15974 nM T41955 C6W9ZE 118719633 IC50 = 23782 nM T41955 C5G1ZL 118719634 IC50 = 2472 nM T41955 CG1L8W 118719635 IC50 = 1562 nM T41955 C9XME2 118719636 IC50 = 18216 nM T41955 C6C9EF 121304827 IC50 > 3000 nM T41955 C1XNR3 121513880 IC50 = 30000 nM T41955 CR3OK6 122178093 IC50 > 10000 nM T41955 CO4U0G 122178094 IC50 = 837 nM T41955 C1VWB3 122178095 IC50 = 951 nM T41955 CX0H4Y 122178096 IC50 = 340 nM T41955 CZ1F4O 122178097 IC50 = 307 nM T41955 C9IJZ7 122178098 IC50 > 6166 nM T41955 C8AJ7G 122178099 IC50 > 7820 nM T41955 CE6NU4 122178100 IC50 > 3249 nM T41955 CNEW07 122178101 IC50 = 1613 nM T41955 CYJ60U 122178102 IC50 > 9356 nM T41955 CTO0H4 122178103 IC50 > 6863 nM T41955 C9NH4L 122178104 IC50 = 288 nM T41955 CW03DO 122178105 IC50 > 10000 nM T41955 C6JPA9 122178106 IC50 = 6104 nM T41955 CRH28X 122178107 IC50 = 190 nM T41955 CA5HR7 122489394 IC50 > 20000 nM T41955 CBD2A5 124086166 EC50 = 3.7 nM T41955 C8EL1W 134014389 EC50 = 39 nM T41955 CR1K3C 134130659 IC50 = 420 nM T41955 C1RBJ4 134132806 IC50 = 59000 nM T41955 CBV0S1 134133658 IC50 = 86000 nM T41955 C29ESF 134133885 IC50 = 2500 nM T41955 CRB8Y9 134145004 IC50 > 100000 nM T41955 C6X8EF 134148902 IC50 > 100000 nM T41955 C65AVS 134153462 IC50 = 9100 nM T41955 C7PN4Y 134154112 IC50 = 10000 nM T41955 CS1U9C 134156923 IC50 = 210 nM T41955 C3TW0A 134374895 IC50 > 30000 nM T41955 CCK5I3 135883253 IC50 = 3 nM T41955 C7IRJ8 137631504 EC50 > 10000 nM T41955 C2L4TX 137631642 EC50 = 3000 nM T41955 CLVS67 137631911 EC50 = 15445 nM T41955 C94QYF 137632127 EC50 = 40000 nM T41955 CC79HI 137632282 EC50 = 1603 nM T41955 CT62IY 137633710 EC50 = 397 nM T41955 CM3S0I 137635409 EC50 = 61 nM T41955 CF1K6B 137635551 EC50 = 900 nM T41955 C2NID5 137637961 EC50 = 1.1 nM T41955 C6B8UI 137639123 EC50 = 52023 nM T41955 CZAF49 137640617 EC50 = 900 nM T41955 CQ6T1L 137641021 EC50 = 63000 nM T41955 C7N0ZA 137642222 EC50 = 400 nM T41955 CT3A7Z 137642393 EC50 = 40 nM T41955 CSN50H 137644695 EC50 = 15955 nM T41955 C45AGL 137645339 EC50 = 21305 nM T41955 CL76KE 137646700 EC50 = 689 nM T41955 CC6RZ1 137647780 EC50 = 236 nM T41955 C7P8DY 137650844 EC50 = 21870 nM T41955 CML5J2 137651080 EC50 = 67 nM T41955 CPR5W1 137653024 EC50 = 21752 nM T41955 C9S4GH 137653297 EC50 = 8000 nM T41955 CG2X5F 137653442 EC50 = 23000 nM T41955 C3K9EZ 137655009 EC50 = 10 nM T41955 C3B8CK 137655606 EC50 = 1813 nM T41955 C5CLY7 137661406 EC50 = 855 nM T41955 CEF8J0 137661941 EC50 = 11000 nM T41955 CNQ0B9 137662053 EC50 = 31146 nM T41955 CEK6B1 139300630 IC50 > 10000 nM T41955 CYKX81 145982566 IC50 > 20000 nM T41955 C76GWJ 145982978 IC50 > 10000 nM T41955 CG5KD2 145983127 IC50 > 10000 nM T41955 COWE81 145984701 IC50 = 390 nM T41955 C28PDY 145984933 IC50 = 109 nM T41955 C5PNL6 145985281 IC50 = 301 nM T41955 CPGE82 145985765 IC50 = 311 nM T41955 CD0T3Z 145986002 IC50 = 1140 nM T41955 CPF95D 155546810 IC50 = 61600 nM T41955 C3AVN9 155554913 IC50 = 18500 nM T41955 D03LVL 53464483 IC50 > 25000 nM T41955 D04AQE 1833 IC50 = 11600 nM T41955 D04NGL 11266244 EC50 = 40 nM T41955 D04ULU 161930 EC50 = 60 nM T41955 D05DAG 164682 IC50 = 13100 nM T41955 D06NGQ 89576 IC50 = 340 nM T41955 D0A1UL 49783953 IC50 = 8.3 nM T41955 D0C8MT 260806 IC50 = 3340 nM T41955 D0D6MC 1150897 IC50 > 30000 nM T41955 D0G8BN 2733484 IC50 = 18000 nM T41955 D0J9CR 16095384 IC50 = 4 nM T41955 D0N7MS 5353376 IC50 = 3900 nM T41955 D0P7VQ 9929425 IC50 = 475 nM T41955 D0Q4GB 637566 EC50 = 5900000 nM T70532 C3W0JR 11379 EC50 = 150000 nM T70532 C96IDF 9855551 EC50 = 90000 nM T70532 C1VQJ2 11195579 EC50 > 500000 nM T70532 CLS28K 11287377 EC50 = 300000 nM T85328 D05EAM 4735 IC50 = 300 nM T85328 CT5E7N 897520 IC50 > 100000 nM T85328 CPQ3D4 1202786 IC50 = 209000 nM T85328 C0QUS5 1618640 IC50 = 14000 nM T85328 CE3S9R 1820399 IC50 > 50000 nM T85328 COGK92 2065762 IC50 = 37200 nM T85328 C9C0OM 2714312 IC50 = 31300 nM T85328 CV9ZH6 2941126 IC50 > 100000 nM T85328 C70MGK 6872119 IC50 > 20000 nM T85328 C85XHT 7509342 IC50 = 56700 nM T85328 CYOS08 8119828 IC50 = 70100 nM T85328 C3NIY8 16456878 IC50 = 209000 nM T85328 CAL45Z 17600651 IC50 = 21000 nM T85328 CWU92E 20866464 IC50 > 50000 nM T85328 CJKO23 20866499 IC50 > 50000 nM T85328 CBXR07 45840460 IC50 = 133200 nM T85328 CEL91T 56923561 IC50 = 89100 nM T85328 C2IT1Z 91383855 IC50 = 170 nM T85328 CU3RP8 124141953 IC50 = 50 nM T85328 C0TE5S 135651612 IC50 = 39800 nM T16738 D0R0MW 5329102 Ki = 6.3 nM T16738 D02XNW 5494449 Ki = 35.8 nM T16738 D03QLG 9917013 IC50 = 114 nM T16738 CWFB78 11305809 IC50 = 1 nM T16738 CRX81Q 71575642 IC50 > 10000 nM T16738 CR72EH 76685062 Ki = 0.17 nM T16738 CZE7X2 78318865 Ki = 110 nM T16738 CNVU13 90292716 Ki = 270 nM T16738 CE38JB 90292741 Ki = 0.4 nM T16738 CV9QD6 145968243 IC50 = 119 nM T16738 D07ADX 54764565 IC50 = 150 nM T16738 D07IHM 9823787 IC50 > 3000 nM T16738 D09QBA 23378546 IC50 > 3000 nM T52297 D0G3PI 449171 EC50 = 1090 nM T52297 D0N0RU 82146 EC50 = 196 nM T52297 D00QWU 59251511 EC50 = 220 nM T52297 D0H4DR 49787490 EC50 = 8 nM T52297 D0L4FS 5280961 IC50 = 31000 nM T52297 D0R9YR 64971 EC50 > 50000 nM T52297 D0S5LT 29435 IC50 > 100000 nM T52297 D04XII 118883505 Ki = 1072 nM T52297 D0TG1V 118883427 Ki = 25 nM T52297 D0W1XE 91827457 Ki = 81 nM T52297 C6RWX2 16260 EC50 = 142 nM T52297 CT52XN 92997 EC50 = 3000 nM T52297 C1BW7P 93017 EC50 > 50000 nM T52297 C1YN4T 121935 EC50 = 470 nM T52297 C5Q7RL 134528 EC50 = 77 nM T52297 CA56RZ 168038 Ki = 180 nM T52297 C5T1DW 644851 EC50 = 526 nM T52297 CXD60C 645748 EC50 = 100 nM T52297 C2EIZ4 680534 IC50 > 30000 nM T52297 CIC0D5 856237 EC50 = 2178 nM T52297 CSHG48 1186353 EC50 = 4000 nM T52297 CZ6Q1Y 1734080 IC50 = 315 nM T52297 C1YK9J 4585579 EC50 = 2468 nM T52297 CO76JI 4730488 EC50 = 309 nM T52297 CF58OK 5188108 EC50 = 100 nM T52297 C54OLI 5288679 EC50 = 50 nM T52297 C16ZSG 6439929 EC50 > 100000 nM T52297 C6R3GO 6539523 EC50 = 1590 nM T52297 C35IYW 8001903 EC50 = 150 nM T52297 C4QM3A 9808622 EC50 = 305 nM T52297 CD3CZ1 9817887 EC50 = 180 nM T52297 COQ43R 9867761 EC50 = 20 nM T52297 CSP19Z 9930940 EC50 = 1300 nM T52297 CL78FK 9953856 EC50 = 600 nM T52297 CI7CS1 10001458 IC50 = 130 nM T52297 CV7SK8 10064801 IC50 = 3100 nM T52297 C3HTA2 10070833 IC50 = 100 nM T52297 C2F4KU 10112384 EC50 = 200 nM T52297 CN24XI 10118997 EC50 = 260 nM T52297 C5NJP2 10129169 EC50 = 46 nM T52297 CG0LQ8 10129170 EC50 = 200 nM T52297 C5VXR7 10135759 EC50 = 220 nM T52297 CF78TR 10143034 EC50 = 250 nM T52297 CQ63JG 10164424 EC50 = 260 nM T52297 C18VCL 10196830 EC50 = 280 nM T52297 CSDA25 10218669 EC50 = 331 nM T52297 CF9PG8 10218693 EC50 = 74 nM T52297 C91PIS 10218694 EC50 = 211 nM T52297 CFA8W3 10230558 EC50 = 660 nM T52297 CHA34M 10231936 EC50 = 45 nM T52297 CWOR09 10252443 EC50 = 140 nM T52297 CL8CU4 10280681 EC50 = 85 nM T52297 C18RJP 10301104 EC50 = 860 nM T52297 CEF95T 10301876 EC50 = 190 nM T52297 C6Q0EM 10312252 EC50 = 365 nM T52297 C0GXN7 10312324 EC50 = 43 nM T52297 C4HDK8 10342621 EC50 = 170 nM T52297 CQ6R0U 10431545 EC50 = 220 nM T52297 CI34YL 10433666 EC50 = 50 nM T52297 CLP71Z 10528213 IC50 = 2000 nM T52297 CQ3US7 10715273 EC50 = 720 nM T52297 CN8I9V 10742556 EC50 = 450 nM T52297 C35FRP 10838864 EC50 = 50 nM T52297 C8RPQ4 11036808 EC50 = 180 nM T52297 C4M1IF 11037703 EC50 = 170 nM T52297 CEG60T 11153463 EC50 = 105 nM T52297 C71EUS 11169139 IC50 = 30.2 nM T52297 C0Q8NA 11180636 EC50 = 63 nM T52297 CI3OJ6 11181120 EC50 = 56 nM T52297 CQGU73 11191949 IC50 = 7 nM T52297 C4DW7B 11261037 IC50 = 130 nM T52297 CK9V6O 11273187 EC50 = 39 nM T52297 C4JS1R 11352536 IC50 = 165 nM T52297 CS25IB 11360909 IC50 = 260 nM T52297 C5XF7R 11377209 EC50 = 20 nM T52297 CPGA59 11489411 EC50 = 23 nM T52297 CRAZ96 11496708 EC50 = 20 nM T52297 C6CR9V 11503359 IC50 = 90 nM T52297 C1ZNO8 11503562 EC50 = 40 nM T52297 C0MX6B 11525365 EC50 = 1100 nM T52297 C68RSH 11525752 IC50 = 18 nM T52297 CEDS09 11555148 EC50 = 510 nM T52297 CXV3T1 11555706 IC50 = 10000 nM T52297 CYS53Q 11559891 IC50 = 2700 nM T52297 CC68LI 11574384 IC50 = 50 nM T52297 C40UZA 11576047 EC50 = 620 nM T52297 C3ITH1 11582802 IC50 = 70 nM T52297 CP53LK 11583743 IC50 = 19 nM T52297 CU0D9H 11584508 IC50 = 6 nM T52297 C7FD2W 11592304 IC50 = 13 nM T52297 C3D7KA 11604995 IC50 = 2000 nM T52297 CK03GD 11611604 IC50 = 6 nM T52297 CX35ZF 11617908 EC50 = 3300 nM T52297 C8EP5Z 11619338 IC50 = 105 nM T52297 CQN62W 11626766 IC50 = 73 nM T52297 C4ZR8D 11627859 IC50 = 9.5 nM T52297 C2WU8Q 11632271 EC50 = 700 nM T52297 C5Y1GK 11633117 IC50 = 20 nM T52297 C0T4UI 11639715 EC50 = 1000 nM T52297 CTW7E6 11655554 IC50 = 180 nM T52297 CN26HX 11655575 EC50 = 3000 nM T52297 CX2H4T 11655676 EC50 = 100 nM T52297 C0N7VQ 11661439 IC50 = 500 nM T52297 CC0PO9 11662127 EC50 = 280 nM T52297 CQ2M8V 11669781 EC50 = 590 nM T52297 C9CQZ7 11683023 IC50 = 3 nM T52297 C47YFZ 11696530 EC50 = 2100 nM T52297 CHW8N7 11697813 EC50 = 6000 nM T52297 CTP37R 11697907 EC50 = 30 nM T52297 CXB9Q8 11698867 IC50 = 5 nM T52297 C7P8FY 11704978 IC50 = 72 nM T52297 CGK13J 11705301 IC50 = 410 nM T52297 C9L7MN 11705887 EC50 = 80 nM T52297 CG4IW2 11713433 EC50 = 300 nM T52297 C0MIV8 11713676 EC50 = 1000 nM T52297 CFRG03 11721039 EC50 = 100 nM T52297 C7VW3O 11813747 EC50 = 85 nM T52297 C3BJQ6 11853545 EC50 = 18100 nM T52297 CJXH73 11853546 IC50 = 1336000 nM T52297 CWFP80 11853793 EC50 = 8410 nM T52297 CPI3X0 11853795 IC50 > 1000000 nM T52297 C9VCA1 11854313 IC50 > 1000000 nM T52297 CQ47XY 11854314 IC50 = 1191000 nM T52297 CBNC08 11854315 IC50 = 62000 nM T52297 CR4W3T 11854316 IC50 = 92000 nM T52297 CM9Q3O 11854570 EC50 = 15300 nM T52297 C4I2NG 11854572 IC50 = 1826000 nM T52297 C5QL6N 11854573 IC50 = 180000 nM T52297 CSN35D 11855081 IC50 = 62000 nM T52297 CS0IL9 11855082 EC50 = 6000 nM T52297 CCJ1N2 11855620 EC50 = 11100 nM T52297 CZ80OQ 11855623 IC50 > 1000000 nM T52297 CMF9T0 11855894 IC50 = 179000 nM T52297 CXZW51 11856960 EC50 = 8320 nM T52297 CGYJ27 11857210 IC50 = 147000 nM T52297 C7HN1R 11857214 IC50 > 1000000 nM T52297 CKS09G 12949989 EC50 = 2202 nM T52297 C2V9RQ 13028610 EC50 = 1189 nM T52297 CG7U2N 14239481 EC50 = 390 nM T52297 CO9C7U 15597289 EC50 = 670 nM T52297 C3HA7T 15953841 IC50 = 955 nM T52297 C43ZTW 16049406 IC50 = 310 nM T52297 CA1U0H 16049407 IC50 = 120 nM T52297 CFMX18 16049474 IC50 = 160 nM T52297 C8ZY3L 16049475 IC50 = 90 nM T52297 CK75FX 16049476 IC50 = 180 nM T52297 CCF48P 16049477 IC50 = 615 nM T52297 C46MDG 16049478 IC50 = 890 nM T52297 CC95QW 16049479 IC50 = 560 nM T52297 CPIM37 16049537 IC50 = 190 nM T52297 CH42EK 16049538 IC50 = 220 nM T52297 CU9G5E 16049539 IC50 = 775 nM T52297 C9D5TB 16049540 IC50 = 195 nM T52297 CEX8N2 16049541 IC50 = 170 nM T52297 CT32VG 16090326 IC50 > 1000 nM T52297 CCT84J 16090327 IC50 = 1871 nM T52297 C03ZSF 16090328 IC50 = 723 nM T52297 C28VIS 16090329 IC50 = 16.5 nM T52297 CF4J1K 16090330 IC50 = 7.6 nM T52297 CUR0Y7 16090331 IC50 = 47 nM T52297 C1IF8A 16090332 IC50 = 274 nM T52297 CL45DA 16718799 IC50 = 115 nM T52297 CKH5O1 16725052 EC50 = 220 nM T52297 C6NOS9 16727104 IC50 = 5.2 nM T52297 CXVS20 16727105 IC50 = 10.2 nM T52297 CN6CU3 16739344 EC50 = 467 nM T52297 C2LMW1 18565134 EC50 = 2600 nM T52297 C0QKH8 18565138 EC50 = 4100 nM T52297 CGS1R9 18565141 EC50 = 3900 nM T52297 CP3AS5 19835803 EC50 = 396 nM T52297 CU4R2K 20704052 EC50 = 10 nM T52297 CL2Y6T 20704053 EC50 = 100 nM T52297 C6OSB4 20704089 EC50 = 2000 nM T52297 CYW1U6 20704115 EC50 = 200 nM T52297 C38JEL 20704150 EC50 = 320 nM T52297 C38ZGD 20704166 EC50 = 1000 nM T52297 CWU4M0 20704168 EC50 = 5000 nM T52297 C6FGV5 20704187 EC50 = 1000 nM T52297 CJTU28 20704188 EC50 = 200 nM T52297 CU1W3Y 20704189 EC50 = 100 nM T52297 CTE9J2 21050637 IC50 > 10000 nM T52297 C1GB2P 21593998 EC50 > 15000 nM T52297 C0FQ7Y 21943462 IC50 = 500 nM T52297 C9MFJ3 21943465 IC50 = 200 nM T52297 CKQ7J8 22042567 IC50 = 1500 nM T52297 CL56EK 22042589 IC50 = 200 nM T52297 CGC2J5 22042622 IC50 > 10000 nM T52297 CPA92E 22042635 IC50 = 400 nM T52297 CWD19A 23643871 EC50 = 608 nM T52297 C5W1QM 23648467 IC50 = 16 nM T52297 CL84DN 23648468 IC50 = 8 nM T52297 CZU9G4 23648469 IC50 = 384 nM T52297 C4J1KP 23648470 IC50 = 150 nM T52297 CF9E7D 23648471 IC50 > 10000 nM T52297 CT50PV 23648472 IC50 = 18 nM T52297 CUTE13 23648473 IC50 = 104 nM T52297 CR1JB8 23648474 IC50 = 650 nM T52297 CX6FT2 23648475 IC50 = 9 nM T52297 CS26KY 23648476 EC50 = 121 nM T52297 CRS43H 23648477 IC50 = 33.6 nM T52297 C6CAG2 23648478 IC50 = 63.9 nM T52297 CFG0L7 23648479 IC50 > 10000 nM T52297 CYA97J 23648480 IC50 = 420 nM T52297 C26XFS 23648481 IC50 = 15.2 nM T52297 CH6O5G 23648482 IC50 = 17.2 nM T52297 CY4I6V 23648483 IC50 = 33.6 nM T52297 C2RJ1K 23648484 IC50 = 11 nM T52297 CO8M2W 23648485 IC50 = 34 nM T52297 CE1G7K 23648486 IC50 = 241 nM T52297 C03PJK 23648487 IC50 = 90.5 nM T52297 CD1N3S 23648488 IC50 = 456 nM T52297 C0RCT4 23648532 EC50 = 346 nM T52297 CG2V6T 23648533 EC50 = 1400 nM T52297 C30RES 23648534 EC50 = 1400 nM T52297 CXOG70 23648535 EC50 = 180 nM T52297 CYL8W7 23648536 EC50 = 70 nM T52297 C9A4RZ 23648537 EC50 = 1900 nM T52297 CJD4H1 23648538 EC50 = 3900 nM T52297 CX5FC4 23648540 EC50 = 6700 nM T52297 C6OM0B 23648541 EC50 = 1500 nM T52297 CA25OJ 23648542 EC50 = 2100 nM T52297 CIDA95 23648543 EC50 = 2400 nM T52297 C1J5LG 23648544 EC50 = 900 nM T52297 CG8J3O 23648545 EC50 = 900 nM T52297 CU7BE2 23648546 EC50 = 700 nM T52297 CTE1N2 24748569 EC50 > 10000 nM T52297 C06CYE 24764397 EC50 = 228 nM T52297 CPJB16 24768116 EC50 = 100 nM T52297 CH58ID 24768117 EC50 = 130 nM T52297 C1ZJT0 24768118 EC50 = 300 nM T52297 CKJ8O1 24768119 EC50 = 275 nM T52297 CR7VX5 24768120 EC50 = 575 nM T52297 C7WA9T 24768121 EC50 = 890 nM T52297 CA52ER 24768122 EC50 = 725 nM T52297 CT2SK4 24768123 EC50 = 5900 nM T52297 CV57AQ 24768125 EC50 = 170 nM T52297 CP0GA4 24808559 EC50 = 1700 nM T52297 C76BPI 24860506 IC50 = 2200 nM T52297 C5PJ0G 24860507 IC50 = 3600 nM T52297 C8C4ME 24860508 IC50 = 25000 nM T52297 C62QOY 24860509 IC50 = 7600 nM T52297 C67AFM 24860510 IC50 = 2500 nM T52297 CV1Q0H 24936142 EC50 = 685 nM T52297 C6ZG0A 24936147 EC50 = 7866 nM T52297 CC13ZW 24936148 IC50 = 745 nM T52297 C18VZL 24986297 EC50 = 2800 nM T52297 CU6Z5R 24986298 EC50 = 2700 nM T52297 CL10IN 24986299 EC50 = 1300 nM T52297 CUV4C0 24986301 EC50 = 1800 nM T52297 CEA64D 24991075 EC50 = 3200 nM T52297 CO08HG 24991077 EC50 = 2200 nM T52297 CFJ34K 24991433 EC50 = 1900 nM T52297 C14HGJ 24991436 EC50 = 2200 nM T52297 CC0QH2 24991785 EC50 = 2500 nM T52297 CF1HS7 24991787 EC50 = 2200 nM T52297 CA1MU6 24991788 EC50 = 2200 nM T52297 CN6J4S 25099837 IC50 = 560 nM T52297 CZW14K 25099838 IC50 = 8.1 nM T52297 CD9W8I 25099839 IC50 = 13 nM T52297 CN97XU 25099842 IC50 = 13.4 nM T52297 CCA5I2 25099990 IC50 = 1.4 nM T52297 CFPR78 25099991 IC50 = 3.2 nM T52297 CE5M6T 25100147 IC50 = 42 nM T52297 CS3ZP8 25100148 IC50 = 8.2 nM T52297 C83EZA 25100149 IC50 = 1.2 nM T52297 CY0V6M 25100150 IC50 = 1 nM T52297 CS87WP 25100151 IC50 = 1.9 nM T52297 CLA0E4 25100152 IC50 = 1.1 nM T52297 CR7EZ5 25100307 IC50 = 3 nM T52297 C4VF6J 25100311 IC50 = 0.92 nM T52297 CBOL78 25100472 IC50 = 2.8 nM T52297 CQSF65 25100922 IC50 = 2.4 nM T52297 CQL7E3 25102117 IC50 = 1.6 nM T52297 CPG4W6 25102118 IC50 = 2.6 nM T52297 C4ANQ0 25102119 IC50 = 1.8 nM T52297 CI4O1G 25102122 IC50 = 8.2 nM T52297 C0QD2M 25102124 IC50 = 6348 nM T52297 C7XW8B 25102125 IC50 = 6.6 nM T52297 CBY8K4 25107513 IC50 = 170 nM T52297 CF1S8P 25132150 IC50 = 4100 nM T52297 C3KC6G 25137978 EC50 = 1810 nM T52297 CO80QT 25137979 EC50 = 5020 nM T52297 C08ANI 25137980 IC50 = 317 nM T52297 C4WMH5 25137981 EC50 = 12770 nM T52297 CG87IF 25137982 IC50 = 260 nM T52297 CU6YO2 25137983 EC50 = 14400 nM T52297 CS3V8P 25137984 EC50 = 15210 nM T52297 C0DX5J 25137985 EC50 = 13440 nM T52297 C87YAR 25137986 EC50 = 15830 nM T52297 CB3CS4 25137987 IC50 = 3101 nM T52297 CB6J0R 25147499 EC50 = 14 nM T52297 CI2XO4 25190753 EC50 = 110 nM T52297 C5TQ2G 25190754 EC50 > 3000 nM T52297 CN67OC 25190755 EC50 = 630 nM T52297 C5B4MW 25190756 EC50 = 226 nM T52297 CWS3O8 25190757 EC50 = 60 nM T52297 C53TOB 25190792 EC50 = 1500 nM T52297 C2P7YG 25190805 EC50 = 1190 nM T52297 CF9EX0 25190808 EC50 = 1150 nM T52297 CHMP24 25190809 EC50 = 1110 nM T52297 CW4DI9 25190847 EC50 = 4300 nM T52297 CX9TD7 25190861 EC50 = 570 nM T52297 CEDZ28 25190863 EC50 = 540 nM T52297 CHS74M 25190864 EC50 > 30000 nM T52297 C8DI4A 25210583 EC50 = 19 nM T52297 C14HCZ 25218828 EC50 = 1600 nM T52297 CM4WA9 25218829 EC50 = 5810 nM T52297 C5U2ED 25218830 EC50 = 5800 nM T52297 C2VFE6 25218831 IC50 = 820 nM T52297 CA0H5N 25218832 IC50 = 540 nM T52297 CE7HR1 25218833 EC50 = 2300 nM T52297 CGY57P 25218834 IC50 = 100 nM T52297 CUP27J 25218835 IC50 = 73 nM T52297 C1D7CS 25218836 EC50 = 1070 nM T52297 CZ09XS 25218837 EC50 = 840 nM T52297 CWHJ63 25218838 IC50 = 49 nM T52297 CBV2X7 25218839 IC50 = 100 nM T52297 CPY79U 25218840 EC50 = 1070 nM T52297 CKX1O5 25218841 EC50 = 2750 nM T52297 CRA4T3 25218842 EC50 = 4230 nM T52297 CF5BR4 25218843 EC50 = 1550 nM T52297 CXN2U4 25218844 EC50 = 1090 nM T52297 C4MWC5 25218845 EC50 = 770 nM T52297 C8W0TY 25218846 IC50 = 920 nM T52297 C7MU6E 25218847 EC50 = 430 nM T52297 CO95WI 25218848 IC50 = 300 nM T52297 CUS41I 25218849 IC50 = 210 nM T52297 CTP8D4 25218850 EC50 = 1260 nM T52297 CVF58N 25218851 EC50 = 370 nM T52297 C0CYW9 25218852 EC50 = 160 nM T52297 C3UI9O 25225010 IC50 = 157 nM T52297 CWO5V0 25225786 IC50 = 11 nM T52297 CZ9CE5 25226691 IC50 = 58 nM T52297 CX3ID9 25226692 IC50 = 161 nM T52297 C9TJ4D 25226881 IC50 = 21 nM T52297 CQIB51 25227069 IC50 = 21 nM T52297 C4Q5BN 25227247 IC50 = 31 nM T52297 CS1EJ7 25234324 EC50 = 2700 nM T52297 C0VHF6 42601437 EC50 = 3400 nM T52297 CR09VW 42641405 EC50 = 20 nM T52297 C5BT2G 42641974 IC50 = 0.8 nM T52297 C53TKQ 44123769 EC50 = 345 nM T52297 C0J5LA 44135945 IC50 = 136 nM T52297 CC41IF 44136012 IC50 = 4.7 nM T52297 CYEQ65 44136014 IC50 = 17 nM T52297 CD5N0Y 44136075 EC50 = 890 nM T52297 CWNG36 44136213 IC50 = 7.5 nM T52297 CP51NL 44136346 IC50 = 89 nM T52297 C4E8PW 44136349 IC50 > 1000 nM T52297 C2V6PL 44136351 IC50 = 194 nM T52297 C9Z3FW 44136417 IC50 = 2.7 nM T52297 CK0WE9 44136418 IC50 = 2.4 nM T52297 C7QRB9 44136419 IC50 = 4 nM T52297 CFI79Y 44136477 EC50 = 540 nM T52297 C4OGJ0 44136604 IC50 = 43 nM T52297 CJM3P2 44136717 EC50 = 710 nM T52297 C9XS4G 44136902 IC50 = 5.7 nM T52297 C3SK9J 44136969 EC50 = 570 nM T52297 CA87MH 44137029 IC50 = 5.4 nM T52297 C41PXG 44137030 IC50 = 38 nM T52297 CAN35S 44137031 IC50 = 13 nM T52297 CD0ET3 44137032 IC50 = 13 nM T52297 CP13OK 44137033 IC50 = 24 nM T52297 CIJA24 44137094 IC50 = 166 nM T52297 C9IXQ3 44137098 IC50 > 1000 nM T52297 C8B9ZN 44137168 IC50 = 1.5 nM T52297 C90LGQ 44137229 IC50 = 292 nM T52297 C0FDZ1 44137303 IC50 = 44 nM T52297 C9QR5C 44137304 IC50 = 1.7 nM T52297 CLTG76 44137366 IC50 = 49 nM T52297 CH8UB0 44137367 IC50 = 30 nM T52297 C9R0KB 44137369 IC50 = 187 nM T52297 CNB45D 44137441 IC50 = 1 nM T52297 C5EL2Q 44137442 IC50 = 1.1 nM T52297 CW41UJ 44137443 IC50 = 4.2 nM T52297 CC9Y5H 44137444 IC50 = 1.2 nM T52297 C86AME 44137503 IC50 = 188 nM T52297 C89GVM 44137575 IC50 = 1.3 nM T52297 C1GH4M 44137576 EC50 = 162 nM T52297 CH50TJ 44137636 EC50 = 420 nM T52297 CW7IY5 44137712 IC50 = 269 nM T52297 C5NFR2 44137713 IC50 = 7.3 nM T52297 C6R1UH 44137714 IC50 = 5.1 nM T52297 CHA73X 44137715 IC50 = 5.6 nM T52297 CF8D0P 44137845 IC50 = 20 nM T52297 CSO53M 44137979 IC50 = 3.7 nM T52297 C28EXH 44137980 IC50 = 3.5 nM T52297 CNVL89 44137982 IC50 = 3.6 nM T52297 CL04IU 44156271 EC50 = 47000 nM T52297 CK8R4C 44180521 IC50 = 68 nM T52297 COEB58 44399795 EC50 = 1 nM T52297 CHT2S3 44400184 IC50 = 90 nM T52297 C1XZ3Q 44400273 EC50 = 320 nM T52297 C2F7JU 44400646 EC50 = 2 nM T52297 C4FA9O 44400680 EC50 ~ 100 nM T52297 C3G2HU 44400748 EC50 = 1 nM T52297 CRWF17 44403557 EC50 = 360 nM T52297 CWT40V 44403558 EC50 = 70 nM T52297 CZT94C 44403564 EC50 = 430 nM T52297 C5XQW3 44403565 EC50 = 150 nM T52297 CD9S3C 44403570 EC50 = 1500 nM T52297 C8K9ZM 44403571 EC50 = 170 nM T52297 C9C2JX 44403589 IC50 = 1670 nM T52297 CTN5Z2 44403617 IC50 = 2800 nM T52297 C34OXW 44403619 EC50 > 50000 nM T52297 C31FVO 44403620 IC50 = 5060 nM T52297 CU4H2G 44403625 IC50 = 3800 nM T52297 C5V6GE 44403626 EC50 = 5200 nM T52297 CA2CW3 44403633 EC50 = 3100 nM T52297 CC7J1B 44403639 EC50 = 240 nM T52297 C38VRQ 44403645 EC50 = 280 nM T52297 COW1B4 44403655 EC50 = 760 nM T52297 CXPJ14 44403656 EC50 = 320 nM T52297 CZK0P5 44409123 EC50 > 5000 nM T52297 CG8SI7 44409143 EC50 = 3000 nM T52297 CWR37I 44409160 EC50 > 5000 nM T52297 C26MRH 44409315 EC50 = 700 nM T52297 C7XFS3 44409322 EC50 = 8 nM T52297 CGY80Q 44409326 EC50 = 50 nM T52297 CUR0D4 44409358 EC50 = 30 nM T52297 CZE6B5 44409361 EC50 = 30 nM T52297 CW9S1K 44411622 IC50 = 372 nM T52297 CNL81R 44411653 IC50 = 39 nM T52297 CW3AV8 44411661 IC50 = 730 nM T52297 C4MAN2 44411789 IC50 = 110 nM T52297 CHW2N5 44411793 IC50 = 6400 nM T52297 CYJ25W 44411810 IC50 = 530 nM T52297 C8FBH9 44411838 IC50 = 630 nM T52297 C4U2SJ 44411842 IC50 = 18 nM T52297 CJF9L1 44411843 EC50 = 8000 nM T52297 CDA4O0 44411976 IC50 = 6400 nM T52297 CX6DN0 44411977 EC50 = 2600 nM T52297 CP46GF 44412005 EC50 = 170 nM T52297 CBVJ21 44412006 IC50 = 60 nM T52297 C8DPK5 44412188 IC50 = 580 nM T52297 CPK6G2 44412195 IC50 = 117 nM T52297 CEU76F 44416756 IC50 = 100 nM T52297 CR97GI 44416799 IC50 = 700 nM T52297 C3YB5A 44416802 IC50 = 1300 nM T52297 CNC6B7 44416803 EC50 = 500 nM T52297 CK82QS 44416818 EC50 = 9400 nM T52297 CZN20F 44416819 EC50 = 10900 nM T52297 C0R2KB 44416821 IC50 = 400 nM T52297 C1SQM3 44416822 EC50 = 1900 nM T52297 CL9HK1 44416842 IC50 = 600 nM T52297 CIXR07 44416843 IC50 = 12000 nM T52297 C6DU1G 44416861 EC50 = 10000 nM T52297 C2GD1Q 44416897 EC50 = 500 nM T52297 CZ1N4K 44416914 IC50 = 200 nM T52297 C4L7VQ 44416915 EC50 = 200 nM T52297 C53BAF 44416930 IC50 = 60 nM T52297 CW3NF9 44416950 IC50 = 1100 nM T52297 CQHE10 44416951 EC50 = 400 nM T52297 CP8Y5T 44416988 EC50 = 9300 nM T52297 C5RB8X 44416991 IC50 = 18000 nM T52297 CDG8Z0 44416992 IC50 = 100 nM T52297 C6MEG2 44417023 EC50 = 2200 nM T52297 CPSL50 44417026 EC50 = 800 nM T52297 CR82JZ 44417027 EC50 = 700 nM T52297 CWDI21 44417028 IC50 = 60 nM T52297 CB6LY0 44417045 IC50 = 5400 nM T52297 CKR1H6 44417046 IC50 = 50 nM T52297 COX48N 44417052 EC50 = 1100 nM T52297 C1TH7E 44417068 IC50 = 50 nM T52297 CAJH47 44417072 IC50 = 100 nM T52297 CL50IQ 44423673 IC50 = 479 nM T52297 CQK4F0 44446235 IC50 = 17 nM T52297 C6E8BG 44446237 IC50 = 112 nM T52297 CGI9W5 44446239 IC50 = 65 nM T52297 CC29YZ 44446242 IC50 = 528 nM T52297 C34HCM 44446244 IC50 = 16 nM T52297 CAK9X2 44446246 IC50 = 6 nM T52297 C65ZXY 44446249 IC50 = 21 nM T52297 CZ2T6A 44446253 IC50 = 147 nM T52297 C6GR7Q 44446254 IC50 = 2 nM T52297 CEDU42 44472980 IC50 = 231 nM T52297 C5OUG9 44472981 IC50 = 75 nM T52297 CTZ48C 44472982 IC50 = 47 nM T52297 C0FJT4 44472983 IC50 = 107 nM T52297 CK3H2I 44472984 IC50 = 36 nM T52297 CO8FG1 44472985 IC50 > 1000 nM T52297 CR0Q7O 44472986 IC50 > 1000 nM T52297 CX18UB 44472987 IC50 = 131 nM T52297 CN30ED 44472988 IC50 = 1002 nM T52297 C41NFW 44472989 IC50 = 59 nM T52297 CI92RZ 44472990 IC50 = 6.6 nM T52297 CO7U1F 44472991 IC50 = 494 nM T52297 CS8EI5 44472992 IC50 = 91 nM T52297 CC3KU9 44472993 IC50 = 74 nM T52297 CZO32E 44472994 IC50 = 12 nM T52297 CTI06D 44472995 IC50 = 12 nM T52297 C69VFJ 44472996 IC50 = 20 nM T52297 CE58LO 44472997 IC50 = 9 nM T52297 C6U0PL 44472998 IC50 = 272 nM T52297 CKB13G 44472999 IC50 = 280 nM T52297 CKOR84 44473000 IC50 = 357 nM T52297 C31XLA 44473001 IC50 = 108 nM T52297 CI7C5U 44473002 IC50 = 34 nM T52297 CFMP64 44473003 IC50 = 50 nM T52297 C01LIU 44473004 EC50 = 1237 nM T52297 CR5SI0 44476535 EC50 > 10000 nM T52297 CDY1W2 44537910 IC50 = 6600 nM T52297 C0OC3N 44559230 EC50 > 50000 nM T52297 CW5RK4 44559244 EC50 > 50000 nM T52297 CEYC85 44564595 EC50 = 480 nM T52297 CV9MX0 44568830 IC50 = 115 nM T52297 CK0TW9 44573589 EC50 = 3300 nM T52297 CJW4Z1 44573631 EC50 = 1820 nM T52297 C2G3FO 44573632 EC50 = 1970 nM T52297 CTOW18 44573633 EC50 = 1000 nM T52297 C18HPE 44573634 EC50 > 30000 nM T52297 CQ97MR 44573677 EC50 = 1080 nM T52297 C3DS6K 44573678 EC50 = 470 nM T52297 CL4G0H 44573679 EC50 = 3100 nM T52297 C89JSN 44573717 EC50 > 30000 nM T52297 C63LBJ 44573718 EC50 = 3500 nM T52297 C2M5UG 44573719 EC50 > 30000 nM T52297 C3YB2D 44626292 EC50 = 9 nM T52297 C4GC8P 45100506 EC50 = 79.43 nM T52297 CA41BS 45270660 IC50 = 668000 nM T52297 C0J3SN 45271480 IC50 = 134000 nM T52297 CR8S4O 45272392 EC50 = 13500 nM T52297 CW79BY 45273240 IC50 = 332000 nM T52297 C3MFY7 45273258 EC50 = 12000 nM T52297 CD9HP7 45481812 IC50 = 5100 nM T52297 CS2UX1 45481813 IC50 = 3900 nM T52297 C3PFR7 45481814 IC50 > 30000 nM T52297 C4YMB1 45481815 IC50 = 4200 nM T52297 CZ8Q5T 45481819 IC50 > 30000 nM T52297 CV21SO 45481820 IC50 = 4800 nM T52297 CJPO37 45481822 IC50 = 8800 nM T52297 C52JWR 45481823 IC50 > 30000 nM T52297 C40FHL 45481824 IC50 = 1700 nM T52297 C47JKF 45481825 IC50 > 3000 nM T52297 C43HEV 45481826 IC50 > 30000 nM T52297 CKT4W8 45481827 IC50 = 2600 nM T52297 C0FZ7X 45481832 IC50 = 3800 nM T52297 CL86HQ 45481833 IC50 = 5500 nM T52297 C9BCY0 45481835 IC50 = 6100 nM T52297 CVZ52U 45481836 IC50 > 30000 nM T52297 C07VHN 45481837 IC50 = 15000 nM T52297 C1EDT6 45481838 IC50 = 2600 nM T52297 CL4XN0 45481843 IC50 = 1600 nM T52297 C4MFG7 45481845 IC50 > 30000 nM T52297 CHSL86 45481846 IC50 > 30000 nM T52297 C0WEA4 45481847 IC50 > 20000 nM T52297 C59QUA 45481848 IC50 = 7400 nM T52297 CTV19K 45481849 IC50 = 9800 nM T52297 C94EIX 45481850 IC50 = 6300 nM T52297 CJ0Z8I 45481851 IC50 = 3700 nM T52297 C0RH7Z 45481853 IC50 = 11000 nM T52297 C7WZ9H 45481854 IC50 > 30000 nM T52297 CFV3R5 45481855 IC50 > 30000 nM T52297 C4ORE2 45481858 IC50 > 30000 nM T52297 C69RLK 45481859 IC50 = 2700 nM T52297 CZE8O5 45481861 IC50 = 6100 nM T52297 C8QNC7 45483602 EC50 = 380 nM T52297 CEF0U7 46186945 IC50 = 165 nM T52297 C4WH5O 46191159 EC50 = 3000 nM T52297 CW76XG 46191160 EC50 = 4500 nM T52297 C0M8HC 46202578 IC50 > 1000 nM T52297 C2M9LX 46202579 IC50 > 1000 nM T52297 CY0B3G 46202580 IC50 > 1000 nM T52297 C35THS 46202902 IC50 > 1000 nM T52297 CA41NL 46202903 IC50 > 1000 nM T52297 C1HP7B 46202904 IC50 > 1000 nM T52297 C6IGM9 46202905 IC50 > 1000 nM T52297 C5LOI9 46202906 IC50 > 1000 nM T52297 CG2K7B 46202907 IC50 = 734 nM T52297 CS12DL 46202929 EC50 = 10 nM T52297 CVKU68 46202930 EC50 = 6.31 nM T52297 C0GOL4 46202931 EC50 = 100 nM T52297 CF5D2Q 46202932 EC50 = 12.59 nM T52297 CV91AT 46203225 IC50 > 1000 nM T52297 C6I3NU 46203226 IC50 > 1000 nM T52297 CY34FM 46203248 EC50 = 79.43 nM T52297 CGF3P7 46203249 EC50 = 125.89 nM T52297 CD0K4Y 46206336 IC50 > 1000 nM T52297 C18TZO 46225114 IC50 > 10000 nM T52297 CQW01V 46225115 IC50 = 6864 nM T52297 C4VBQ8 46225151 IC50 = 26613 nM T52297 C1M2NC 46225152 IC50 = 445 nM T52297 CB94AX 46225194 IC50 = 29850 nM T52297 CZL91B 46225195 IC50 = 552 nM T52297 C8P3HN 46225196 IC50 = 1770 nM T52297 CZ7K6G 46225197 IC50 = 453 nM T52297 C9FD3L 46225243 IC50 = 1365 nM T52297 CQ94OV 46225244 IC50 = 286 nM T52297 C2R5PZ 46225245 IC50 = 756 nM T52297 CO56AF 46225246 IC50 = 12700 nM T52297 CE2W0C 46225296 IC50 > 10000 nM T52297 CN9JT0 46226318 EC50 = 700 nM T52297 CT3E5K 46226367 IC50 > 1000 nM T52297 C4KVS8 46226434 EC50 = 1570 nM T52297 C4NM1R 46226975 IC50 = 7.2 nM T52297 CR6X9K 46877573 EC50 = 950 nM T52297 C4QTV3 46877575 IC50 = 279 nM T52297 C9LQM2 46877576 IC50 = 69 nM T52297 C9DVO7 46877577 IC50 = 2 nM T52297 C0YDO7 46877578 IC50 = 30 nM T52297 COJN09 46887743 IC50 > 1000 nM T52297 C0Q8VO 46887744 IC50 = 9 nM T52297 CJW63M 46887745 IC50 > 1000 nM T52297 C0PK3A 46887797 IC50 = 7 nM T52297 CQCD45 46887798 IC50 = 372 nM T52297 CM23GQ 46887799 IC50 = 4.8 nM T52297 CCG9X7 46887800 IC50 = 7.6 nM T52297 CK41YM 46887851 IC50 = 8.2 nM T52297 CFY72K 46887852 IC50 = 362 nM T52297 CDPU51 46887853 IC50 = 73 nM T52297 C1D6VN 46887854 IC50 = 12 nM T52297 C3ZMN8 46887888 IC50 > 1000 nM T52297 C8BLU0 46887889 IC50 = 10 nM T52297 COL94T 46887890 IC50 = 10 nM T52297 CYI8F3 46887891 IC50 = 32 nM T52297 CVX9L5 46887924 IC50 = 25 nM T52297 CN9L7G 46916268 EC50 > 8300 nM T52297 CP56CJ 49821979 EC50 = 130 nM T52297 C3HQK9 49821981 EC50 = 8 nM T52297 C4LZ1T 49822063 EC50 = 12 nM T52297 CPT4Z8 49822066 EC50 = 69 nM T52297 CIJ50V 49822147 EC50 = 57 nM T52297 CMPO56 49822148 EC50 = 30 nM T52297 CG6LI3 49822225 EC50 = 72 nM T52297 C5CG6O 49822226 EC50 = 11 nM T52297 CUD91T 49862248 EC50 > 10000 nM T52297 C6BM3N 50916706 IC50 > 100000 nM T52297 C2NJ3B 51003508 EC50 = 41000 nM T52297 CM7BY6 53385590 IC50 = 10000 nM T52297 CL78UE 54344821 EC50 = 1500 nM T52297 C5ZX4B 54597874 EC50 > 10000 nM T52297 CUT56J 56589730 EC50 = 1100 nM T52297 CGF2A0 57394020 IC50 = 6300 nM T52297 CTD0E1 57394021 IC50 = 13000 nM T52297 C7DQ1X 57404459 IC50 = 800 nM T52297 CFVN93 57757122 EC50 = 540 nM T52297 C4BTN7 57900760 EC50 = 1700 nM T52297 C9XA5G 57900823 EC50 = 2200 nM T52297 CENS58 57962786 EC50 = 2400 nM T52297 C9PD2F 57962932 EC50 = 2600 nM T52297 C63ZOK 57962935 EC50 = 1500 nM T52297 C6Q5TV 57962956 EC50 = 11000 nM T52297 C8CY6K 57963018 EC50 = 1700 nM T52297 CU6Z4C 59200977 EC50 = 3140 nM T52297 C9VZN3 59200986 EC50 = 2890 nM T52297 C2HYE6 59201075 EC50 = 1960 nM T52297 C0OD8R 59201087 EC50 = 340 nM T52297 CRJ3Q2 59201115 EC50 = 200 nM T52297 C8EB3H 59201131 EC50 = 360 nM T52297 CHLR48 59234874 EC50 = 2800 nM T52297 C73CIF 59234887 EC50 = 1800 nM T52297 CH78VI 59234921 EC50 = 600 nM T52297 CIB7H4 59234952 EC50 = 2400 nM T52297 CE9J7G 59234955 EC50 = 2300 nM T52297 CT8QH0 59234958 EC50 = 500 nM T52297 CSF58L 59234986 EC50 = 860 nM T52297 C2B4OJ 59234998 EC50 = 1700 nM T52297 C2YS3R 59234999 EC50 = 1800 nM T52297 C8E3TC 59235012 EC50 = 710 nM T52297 C6R0AK 59235049 EC50 = 2300 nM T52297 C7F5KX 59235054 EC50 = 1500 nM T52297 CJUK93 59235080 EC50 = 1200 nM T52297 C1E4JW 59235082 EC50 = 900 nM T52297 C84TQU 59235084 EC50 = 1200 nM T52297 CK1JR4 59235110 EC50 = 1400 nM T52297 CK08IO 59235130 EC50 = 400 nM T52297 C3QE7W 59235136 EC50 = 1200 nM T52297 CTO4C0 59235143 EC50 = 1600 nM T52297 CEQD45 59235170 EC50 = 1500 nM T52297 C92RGU 59251295 EC50 = 52 nM T52297 CES06G 59251431 EC50 > 10000 nM T52297 CG2NL0 59251456 EC50 = 200 nM T52297 CU02IZ 59251553 EC50 = 85 nM T52297 C17SAE 59251574 EC50 = 100 nM T52297 C17AXL 59251592 EC50 > 10000 nM T52297 C36TYG 59631866 EC50 = 540 nM T52297 C4LTZ9 59631939 EC50 = 65 nM T52297 CN15OH 59632480 EC50 = 220 nM T52297 CE1K9L 59632482 EC50 = 140 nM T52297 CUVR29 59632565 EC50 = 120 nM T52297 CAKQ02 59633156 EC50 = 320 nM T52297 CJ36PA 59726531 EC50 = 4 nM T52297 CKO07V 61343280 EC50 = 108 nM T52297 CPAB97 61352587 EC50 = 390 nM T52297 CD76EJ 61353182 EC50 = 164 nM T52297 C5H6NQ 66797441 EC50 = 570 nM T52297 CS41OX 67119337 EC50 = 1300 nM T52297 CP1M5T 68655604 EC50 = 18 nM T52297 C5B7DK 71451721 IC50 = 2200 nM T52297 C4WVB2 71451730 IC50 > 10000 nM T52297 C2J0LM 71451731 IC50 > 10000 nM T52297 CM6Z3K 71455271 EC50 = 4200 nM T52297 CGJ60X 71455272 IC50 > 30000 nM T52297 CGE0M4 71457060 IC50 = 19000 nM T52297 CEO4U2 71457061 IC50 = 4900 nM T52297 CTY76D 71457062 EC50 = 910 nM T52297 CP50ZQ 71458918 IC50 = 3500 nM T52297 C3YL4V 71458919 IC50 = 14000 nM T52297 CDM21R 71460722 IC50 = 1300 nM T52297 C8UKI7 71460723 IC50 = 21000 nM T52297 CQU5I1 71460728 IC50 > 30000 nM T52297 C1C3OQ 71460729 IC50 > 30000 nM T52297 C8JXP0 71462452 IC50 = 6100 nM T52297 C9Z2MA 71462453 IC50 > 10000 nM T52297 CPS62O 71462454 EC50 = 1700 nM T52297 CZ9E2O 71462455 IC50 = 1700 nM T52297 CT47LS 71462456 IC50 = 5400 nM T52297 CXK08C 71612420 EC50 = 9200 nM T52297 C1DR8E 71622396 EC50 = 2300 nM T52297 C70QOT 71682479 IC50 = 63000 nM T52297 CAR09D 71682481 IC50 = 20000 nM T52297 C1TB8G 71682483 IC50 = 16000 nM T52297 C4SV3Z 71682624 IC50 = 13000 nM T52297 C6MQ7J 71682626 IC50 = 40000 nM T52297 CL04WU 71682627 IC50 = 40000 nM T52297 CF0Y4S 71682629 IC50 = 32000 nM T52297 C5O9HB 71682631 IC50 = 25000 nM T52297 C6F8IQ 71682633 IC50 = 32000 nM T52297 CBF79Z 71682784 IC50 = 10000 nM T52297 CSJQ97 71682786 IC50 = 16000 nM T52297 C0B1QU 71682787 IC50 = 20000 nM T52297 CACO06 71682788 IC50 = 32000 nM T52297 CQ39RJ 71682789 IC50 = 40000 nM T52297 C5M2FV 71682790 IC50 = 40000 nM T52297 CAV4K9 71682791 IC50 = 50000 nM T52297 CE8TN9 71682936 IC50 > 100000 nM T52297 C7ZLE2 71682938 IC50 = 16000 nM T52297 C0IQ5Y 71682939 IC50 > 100000 nM T52297 CV96CP 71682940 IC50 = 6300 nM T52297 C8C3DJ 71682941 IC50 = 32000 nM T52297 C4KZ9W 72529513 EC50 = 400 nM T52297 CMZ85K 72722807 EC50 > 10000 nM T52297 C2BQO3 72722945 EC50 = 719 nM T52297 C6UWO5 74762670 EC50 > 10000 nM T52297 CJXG25 76284182 EC50 > 10000 nM T52297 CMW6O1 77620538 EC50 = 3700 nM T52297 C7ZMD9 78319220 IC50 > 3000 nM T52297 CV64IH 86233643 EC50 = 1705 nM T52297 C4SA8H 86302482 EC50 > 10000 nM T52297 CBI06J 86346645 EC50 > 10000 nM T52297 C5VCM4 86690644 EC50 > 10000 nM T52297 CGFW70 86690646 EC50 > 10000 nM T52297 C5J9MZ 87123143 EC50 = 1230 nM T52297 CGA6W0 87123160 EC50 = 2000 nM T52297 CB4Y0Z 87198339 EC50 = 3740 nM T52297 C5MOV2 89659415 EC50 > 10000 nM T52297 CLW3O5 89665055 EC50 = 3600 nM T52297 C7E5RV 90200534 EC50 > 10000 nM T52297 CS53WO 91663364 EC50 = 790 nM T52297 CI92WR 91664317 EC50 > 10000 nM T52297 CI0J1E 91827511 EC50 = 310 nM T52297 CT3K8B 117940657 EC50 = 1030 nM T52297 C9R5HF 117949985 EC50 > 7500 nM T52297 C0W6MZ 117950226 EC50 = 315 nM T52297 C39DHO 117951324 EC50 = 99 nM T52297 C4S9EM 117964962 EC50 > 10000 nM T52297 CS4GJ9 117964973 EC50 > 10000 nM T52297 CDXK37 117964975 EC50 > 10000 nM T52297 CN6RT8 117964978 EC50 > 10000 nM T52297 C96BSK 117964998 EC50 > 10000 nM T52297 CW27MY 118063735 EC50 > 10000 nM T52297 C79IOD 118207841 EC50 > 7500 nM T52297 CW27ZE 118207854 EC50 > 3750 nM T52297 C2FLM1 118207907 EC50 > 7500 nM T52297 CXW5M0 118207954 EC50 > 7500 nM T52297 C9UK5A 118207966 EC50 > 7500 nM T52297 C0SQH5 118207970 EC50 > 7500 nM T52297 C0PWH6 118207991 EC50 > 7500 nM T52297 C2U3TJ 118208018 EC50 > 7500 nM T52297 C1MOT7 118208026 EC50 > 7500 nM T52297 CZ2C3U 118208048 EC50 > 7500 nM T52297 CI86YW 118208079 EC50 = 2920 nM T52297 C2KAR6 118208086 EC50 > 7500 nM T52297 C3TJY2 118208092 EC50 > 7500 nM T52297 CS2F1K 118208112 EC50 > 7500 nM T52297 C8N2PF 118208184 EC50 > 7500 nM T52297 C51XTL 118217548 EC50 > 7500 nM T52297 C1FL5I 118217550 EC50 > 7500 nM T52297 CEN76C 118217555 EC50 > 7500 nM T52297 CYRF01 118217561 EC50 = 408 nM T52297 C2LIW9 118217576 EC50 > 7500 nM T52297 CH9T1O 118217580 EC50 > 7500 nM T52297 CIT31Q 118217593 EC50 > 7500 nM T52297 C1ZRN9 118217594 EC50 > 7500 nM T52297 CAUT58 118217595 EC50 > 7500 nM T52297 CB3KO0 118217596 EC50 > 7500 nM T52297 C95ERM 118217608 EC50 > 7500 nM T52297 CM2U4C 118217609 EC50 > 7500 nM T52297 C9V0ZM 118217611 EC50 > 7500 nM T52297 CZ5L3N 118217612 EC50 > 7500 nM T52297 CCK3J9 118217851 EC50 > 7500 nM T52297 CO5I3V 118217852 EC50 > 7500 nM T52297 CD5TJ3 118217853 EC50 > 7500 nM T52297 C6HSC3 118217854 EC50 > 7500 nM T52297 CEKH57 118217858 EC50 > 7500 nM T52297 C1CTB6 118217859 EC50 > 7500 nM T52297 C7U0XR 118217863 EC50 > 7500 nM T52297 CDP0H5 118217865 EC50 > 7500 nM T52297 C82YDU 118217866 EC50 > 7500 nM T52297 CQ60HK 118217867 EC50 > 7500 nM T52297 C9N7VY 118217868 EC50 > 7500 nM T52297 C6LC7H 118217869 EC50 > 7500 nM T52297 CV9G4S 118217870 EC50 > 7500 nM T52297 C8PR3G 118217871 EC50 > 7500 nM T52297 CZ3FX6 118217874 EC50 > 7500 nM T52297 CK85HV 118217875 EC50 > 7500 nM T52297 CT0DV4 118217911 EC50 > 7500 nM T52297 C1QPW5 118217915 EC50 > 7500 nM T52297 C3YTM2 118217920 EC50 > 7500 nM T52297 CU0T7K 118217922 EC50 > 7500 nM T52297 C0ETA2 118217925 EC50 > 7500 nM T52297 C89EDG 118217927 EC50 > 7500 nM T52297 C81QMJ 118217932 EC50 > 7500 nM T52297 C6X4IN 118217935 EC50 > 7500 nM T52297 CD01CA 118526849 EC50 > 10000 nM T52297 CBZ75K 118724654 EC50 > 10000 nM T52297 CAT4B6 118729956 EC50 = 2600 nM T52297 CU08LA 118796406 EC50 = 6930 nM T52297 CQNI87 118883423 Ki = 3 nM T52297 CP75LI 118883429 Ki = 146 nM T52297 CB6F8J 118883492 Ki = 157 nM T52297 CY29BV 118987028 EC50 = 420 nM T52297 C3RFZ1 121596966 Ki = 63 nM T52297 CP52DJ 121596967 Ki = 136 nM T52297 CWV50E 122181445 EC50 = 2400 nM T52297 CRY8N5 122190169 EC50 = 4200 nM T52297 CR20QT 122192261 IC50 > 30000 nM T52297 C9QF1B 122192262 IC50 > 30000 nM T52297 C34OXY 122192263 IC50 > 30000 nM T52297 CE76CW 122192264 IC50 > 30000 nM T52297 CN0D3U 122192265 IC50 > 30000 nM T52297 C3C2MX 122192266 IC50 = 27000 nM T52297 CSHD20 122192267 IC50 > 30000 nM T52297 CHDI48 122192268 IC50 = 23000 nM T52297 CF5Q8I 122192269 IC50 > 30000 nM T52297 C6MEU5 122192270 IC50 = 6800 nM T52297 C58SCX 122192271 IC50 = 30000 nM T52297 C53ACS 122192272 IC50 = 30000 nM T52297 CLJ7S1 122192273 IC50 = 3300 nM T52297 C4UO8G 122192274 IC50 = 13000 nM T52297 CZ6X9G 122192275 IC50 > 30000 nM T52297 CPI25Z 122192276 IC50 = 17000 nM T52297 C8E9GN 122192277 IC50 = 22000 nM T52297 CJ30NY 122192278 IC50 = 25000 nM T52297 CP2X8L 122192279 IC50 > 30000 nM T52297 C80QHL 122192280 IC50 > 30000 nM T52297 C4F9ZK 122669103 IC50 > 10000 nM T52297 CZH39M 122669106 IC50 > 10000 nM T52297 C0T8FO 122669173 IC50 > 10000 nM T52297 CD6X5P 122669265 EC50 > 7500 nM T52297 C0S7UB 122678562 IC50 > 10000 nM T52297 CY8S1P 122678563 IC50 > 10000 nM T52297 C0MUW2 122678576 IC50 > 10000 nM T52297 C2SQ9M 122678748 IC50 > 10000 nM T52297 CH1J6K 122678779 IC50 > 10000 nM T52297 CD9HN3 122678983 IC50 > 10000 nM T52297 CF39TE 122679031 IC50 > 10000 nM T52297 CW37BU 127044455 EC50 = 280 nM T52297 CYO9Q7 127044456 EC50 = 41 nM T52297 C1L5VC 127044605 EC50 = 500 nM T52297 C9QO3M 127044780 EC50 = 2000 nM T52297 CW46GA 127049311 EC50 > 20000 nM T52297 CZW30P 127049312 Ki = 1100 nM T52297 CKM23U 127049313 Ki = 43 nM T52297 CB1IR7 127051155 Ki = 2200 nM T52297 C8JW1U 129167185 EC50 = 163 nM T52297 CB62QX 131953519 EC50 = 2820 nM T52297 CK0G6A 134131424 Ki = 383 nM T52297 CES87G 134135247 Ki = 7 nM T52297 C2A7CZ 134138904 Ki = 204 nM T52297 CBSF46 134142531 EC50 = 110 nM T52297 C8MAB7 134142736 Ki = 86 nM T52297 CVC1Y4 134142943 Ki = 22 nM T52297 CK13YN 134145788 Ki = 48 nM T52297 CR0OX5 134146533 EC50 = 76 nM T52297 CB39QU 134150059 EC50 = 120 nM T52297 C9NI7K 134151534 Ki = 71 nM T52297 CZH50T 134151855 Ki = 51 nM T52297 C0LGI2 134154676 Ki = 20 nM T52297 CZV9B3 134154775 Ki = 186 nM T52297 CJ0UG1 134155310 Ki = 218 nM T52297 CNS38M 134157776 Ki = 32 nM T52297 C1DTF0 137634167 EC50 = 3200 nM T52297 C7R8XI 137635446 EC50 = 16430 nM T52297 C7O1SF 137637681 EC50 = 8510 nM T52297 CN40KU 137638307 EC50 = 1500 nM T52297 CF35PX 137640942 EC50 = 5580 nM T52297 CL79RE 137641742 EC50 = 15750 nM T52297 C6PSI1 137641894 EC50 = 2090 nM T52297 C5W2UL 137643175 EC50 = 6610 nM T52297 CE21KT 137651926 EC50 = 14510 nM T52297 C2V3BP 137657515 EC50 = 8070 nM T52297 CXQ9V8 137659428 EC50 = 4110 nM T52297 CK3X1N 137796283 EC50 > 30000 nM T52297 CC2BH9 145232219 EC50 > 30000 nM T52297 C8BY3E 145720949 EC50 = 15000 nM T52297 CO26VY 145720950 EC50 = 15000 nM T52297 CYD4E5 145720951 EC50 = 16000 nM T52297 CO95TZ 145720952 EC50 = 50000 nM T52297 C79LGM 145720953 EC50 = 5100 nM T52297 C0A8WM 145720954 EC50 = 5300 nM T52297 CSC3F1 145720955 EC50 = 1700 nM T52297 C6NQ9I 145720956 EC50 = 1700 nM T52297 CW3Y0H 145949340 IC50 > 20000 nM T52297 CPK5U1 145951022 IC50 > 20000 nM T52297 CKT24R 145951943 IC50 > 20000 nM T52297 CZM2D7 145963820 EC50 = 70 nM T52297 CI3TP7 145964673 EC50 = 2403 nM T52297 CFK0H4 145965098 EC50 = 265 nM T52297 CKL63D 145965344 EC50 = 3280 nM T52297 C3GI6D 145965669 EC50 = 1300 nM T52297 C4TL7G 145965870 EC50 = 342 nM T52297 C4H9UY 145966156 EC50 = 190 nM T52297 C4P3DR 145967002 EC50 = 970 nM T52297 CY1X5Q 145968478 EC50 > 7500 nM T52297 CG27VL 145969403 EC50 = 374 nM T52297 CYT8M9 145971562 EC50 = 2770 nM T52297 CC8HN9 145973516 EC50 = 2070 nM T52297 C0X3EB 145974156 EC50 > 7500 nM T52297 C13TQJ 145974494 EC50 = 385 nM T52297 CAYQ72 145974767 EC50 = 250 nM T52297 C4SPY0 145974975 EC50 = 40.4 nM T52297 C60CDE 145975835 EC50 = 320 nM T52297 CA3XR1 145976113 EC50 = 980 nM T52297 CQZ7I9 145977465 EC50 = 310 nM T52297 CE2O1P 145977892 EC50 = 290 nM T52297 CB70AE 145980094 EC50 > 30000 nM T52297 CT18YC 145982460 EC50 = 230 nM T52297 CRTG03 145987785 EC50 > 30000 nM T52297 CC89OI 148034311 IC50 > 10000 nM T52297 CE6V8Z 155511797 IC50 > 10000 nM T52297 C9D7ZE 155515113 EC50 = 701 nM T52297 C14OPD 155516918 EC50 = 570 nM T52297 C6SBY9 155521216 EC50 = 115 nM T52297 CU5Z8T 155522788 IC50 > 10000 nM T52297 C1DT9M 155525669 IC50 > 10000 nM T52297 CXS9T8 155526989 IC50 > 10000 nM T52297 C59SQP 155528665 EC50 = 903 nM T52297 CO9N5H 155530678 IC50 > 10000 nM T52297 CIUA10 155537856 IC50 > 10000 nM T52297 CLO98T 155539150 EC50 > 7500 nM T52297 CX97BV 155539638 EC50 = 2285 nM T52297 CDU60J 155539858 EC50 = 5025 nM T52297 CY4OQ3 155541483 EC50 = 2237 nM T52297 C0V6EY 155543172 IC50 > 10000 nM T52297 CX7L0S 155544387 IC50 > 10000 nM T52297 CSK20E 155544524 IC50 > 10000 nM T52297 CTEC81 155544796 EC50 > 7500 nM T52297 CU6DW5 155554454 EC50 = 2470 nM T52297 CBK1E5 155556708 IC50 > 10000 nM T52297 CH62VW 155557200 EC50 = 2130 nM T52297 C3FI7U 155560819 IC50 > 10000 nM T52297 CA91EM 155564933 IC50 > 10000 nM T52297 CPF42S 155565257 IC50 > 10000 nM T52297 C1AJO9 155568648 EC50 = 113 nM T52297 D00DLU 16049480 EC50 = 3000 nM T52297 D00HVP 10070992 IC50 = 4900 nM T52297 D02UID 16734800 IC50 = 179 nM T52297 D06OVX 65094 EC50 = 1160 nM T52297 D06VRA 24860515 IC50 = 3200 nM T52297 D07IZG 50905018 IC50 = 5000 nM T52297 D07XLQ 44537911 IC50 = 200 nM T52297 D08QXD 9935197 EC50 = 35 nM T52297 D08URT 121948 EC50 = 130 nM T52297 D09UND 24860514 IC50 = 5700 nM T52297 D09VLE 24860516 IC50 = 7100 nM T52297 D0A1WR 71478195 IC50 = 214 nM T52297 D0B5FC 447912 EC50 = 3.2 nM T52297 D0C6QI 9830426 EC50 = 1 nM T52297 D0H2YM 123976 EC50 = 250 nM T52297 D0HA0U 24860512 IC50 = 4400 nM T52297 D0IZ9O 24860513 IC50 = 8400 nM T52297 D0K4GK 167685 EC50 = 325 nM T52297 D0L1CX 45481863 IC50 = 7500 nM T52297 D0PL4F 447905 EC50 = 22 nM T52297 D0Q2RP 3247059 EC50 = 95 nM T52297 D0R8LN 45481844 IC50 = 2400 nM T52297 D0U4TN 10638446 IC50 = 13000 nM T52297 D0V3PG 128861 EC50 = 3500 nM T52297 D0V4RZ 25113722 IC50 = 248 nM T52297 D0X2HK 45481821 IC50 = 2900 nM T52297 D0X5DT 10616182 IC50 = 9800 nM T52297 D0Z8LE 24860511 IC50 = 6600 nM T52297 D0Z8RH 25137977 EC50 = 4270 nM T75152 D0X5SD 3117 IC50 = 320 nM T75152 C49BCY 1570 IC50 = 33000 nM T75152 CZ7IA3 1647 IC50 = 550 nM T75152 CKC31Q 86633 IC50 = 2600 nM T75152 C4ZB8R 245718 IC50 = 75000 nM T75152 C39MKT 712750 IC50 = 35000 nM T75152 COB3T1 2132963 IC50 = 5000 nM T75152 CF2N8O 2794167 IC50 = 5910 nM T75152 C94LDM 6459851 IC50 = 91000 nM T75152 C62ZIW 10176672 IC50 = 30000 nM T75152 C9C6LU 10334080 IC50 = 100000 nM T75152 CCUJ60 10445232 IC50 > 1000000 nM T75152 CY41LT 10445774 IC50 > 1000000 nM T75152 CPIV30 13194096 IC50 > 100000 nM T75152 CW1FA3 16227983 IC50 = 16000 nM T75152 CBZP95 16780874 IC50 = 34000 nM T75152 CMO3B7 29130197 IC50 > 100000 nM T75152 CC9VJ0 39047495 IC50 = 50000 nM T75152 CO6A3U 44387955 IC50 = 100000 nM T75152 C3PTZ7 70700688 IC50 = 54000 nM T75152 C3UBY0 122163387 IC50 = 8700 nM T75152 C4P9JW 122516179 IC50 = 2800 nM T75152 CYT3P6 122516185 IC50 = 7300 nM T75152 CMB23H 122516211 IC50 = 3100 nM T75152 CV25IT 122516222 IC50 = 2900 nM T75152 CU9N2M 122516246 IC50 = 5500 nM T75152 CN3VC8 122516255 IC50 = 2400 nM T75152 C4M3ZK 122516295 IC50 = 3100 nM T75152 C4ELG0 122516336 IC50 = 1800 nM T75152 C9BL6C 122516346 IC50 = 8400 nM T75152 CX3B4R 122516830 IC50 = 83000 nM T75152 C41DZW 122516838 IC50 = 93000 nM T75152 COK0J3 122516959 IC50 = 11000 nM T75152 C0AQW4 122517020 IC50 > 100000 nM T75152 CL3Q9Z 122517043 IC50 = 18000 nM T75152 C84UJE 130302628 IC50 = 1260 nM T75152 CL74FP 132253032 IC50 = 30000 nM T75152 CSEW98 132253084 IC50 = 35000 nM T75152 CG6KP2 132253106 IC50 = 21000 nM T75152 CCL91Y 132253144 IC50 = 23000 nM T75152 C4C6HK 132253151 IC50 = 22000 nM T75152 CJAN-32 132253163 IC50 = 16000 nM T75152 CC89LI 132253175 IC50 = 11000 nM T75152 CS0LC7 134280641 IC50 = 16000 nM T75152 CGN6E7 135492608 IC50 = 9200 nM T75152 CC35GR 135615984 IC50 = 1600 nM T75152 CE9O8V 137634616 IC50 = 45000 nM T75152 CI1Y2F 137648233 IC50 = 3500 nM T75152 CTA4O6 137656044 IC50 = 52000 nM T75152 D02UVS 5455 IC50 = 1040 nM T37510 CT31GY 1070501 IC50 = 3800 nM T37510 CZD3A0 1255990 IC50 = 14070 nM T37510 C5DP1O 1306479 IC50 = 15710 nM T37510 CU81GL 1369880 IC50 = 8550 nM T37510 CMUC37 1977212 IC50 = 4800 nM T37510 CZ7N5A 2283538 IC50 = 38050 nM T37510 C0S7DA 5737576 IC50 = 2500 nM T37510 C31QAL 10143532 Ki = 15000 nM T37510 C7VH6K 15950345 Ki = 5700 nM T37510 CRX19I 23646295 Ki = 13000 nM T37510 D02AVL 18376720 Ki > 5000 nM T37510 D02PAU 16731825 Ki > 10000 nM T37510 D0ON2Z 204102 Ki = 19700 nM T37510 D0R9CH 3400921 Ki > 10000 nM T72168 D04DJN 10635 IC50 = 360 nM T72168 D07BSQ 5994 IC50 = 14 nM T72168 D0D1SG 5755 EC50 = 0.002 nM T72168 D0EP0C 5833 IC50 = 1.6 nM T72168 D0G8BV 6450278 Ki = 37 nM T72168 D0I1LH 5839 EC50 = 0.18 nM T72168 D0IT2G 5743 Ki = 0.36 nM T72168 D0Q4SD 443872 IC50 = 63.1 nM T72168 D0Y7IU 5281004 EC50 = 4.8 nM T72168 D0Y7JU 9854489 IC50 = 166 nM T72168 D0Z4EI 55245 IC50 = 590 nM T72168 D00JFE 56941241 IC50 > 1000 nM T72168 D01SYU 10026128 IC50 = 10000 nM T72168 D05RZE 42636651 Ki = 0.33 nM T72168 D07MON 5311505 IC50 = 470 nM T72168 D0SZ1G 121248172 IC50 > 38000 nM T72168 D0X9YP 67041274 IC50 > 10000 nM T72168 D0TH6M 25204767 EC50 > 10000 nM T72168 D0W1XE 91827457 IC50 > 10000 nM T72168 D02KAU 46871935 IC50 = 9 nM T72168 D03KTE 16750192 Ki > 10000 nM T72168 D09UFV 24825740 IC50 > 5000 nM T72168 D0W5RL 9577221 IC50 = 1600 nM T72168 C59UQE 6279 IC50 = 1197 nM T72168 C2O8KM 101788 EC50 = 50 nM T72168 C40YBS 444036 IC50 = 149 nM T72168 C8AMD7 2848661 IC50 = 460 nM T72168 CLBV35 3699263 IC50 = 850 nM T72168 C43BVE 3816305 IC50 = 1070 nM T72168 CDCK27 5185174 IC50 = 1400 nM T72168 C16ZSG 6439929 Ki = 39 nM T72168 C7REX1 9805004 IC50 = 38 nM T72168 CV87EA 9820084 IC50 = 290 nM T72168 C8A3WG 9820510 Ki > 10000 nM T72168 C06RXB 9821393 Ki = 1682 nM T72168 CD9S5P 9825465 Ki = 3838 nM T72168 CE62WD 9839013 IC50 > 1000 nM T72168 CBS8M2 9839134 IC50 = 2369 nM T72168 C92CPK 9841404 Ki > 10000 nM T72168 CK7UC3 9841413 Ki > 10000 nM T72168 C7P6XH 9842832 Ki > 10000 nM T72168 C7RS9U 9846657 Ki > 5000 nM T72168 CERF28 9861044 Ki > 10000 nM T72168 C3K4EU 9862027 Ki > 10000 nM T72168 CEM27C 9885473 IC50 = 3000 nM T72168 C6B9CZ 9888873 IC50 = 160 nM T72168 CZ5R9B 9890023 Ki = 493 nM T72168 CJ7U3R 9904286 IC50 > 10000 nM T72168 C6SWK1 9904610 IC50 = 2492 nM T72168 CTI1J8 9905296 Ki > 10000 nM T72168 CE1TK2 9908041 IC50 > 10000 nM T72168 CMJG42 9921530 IC50 > 10000 nM T72168 C39EXP 9933936 IC50 = 454 nM T72168 C24FUO 9943699 IC50 = 1386 nM T72168 CCSX75 9949772 IC50 = 1500 nM T72168 CKU64T 9952569 IC50 = 333 nM T72168 CW0ED9 9953456 IC50 = 681 nM T72168 C95CAN 9978625 Ki = 0.967 nM T72168 C1QP8T 9993897 IC50 = 2000 nM T72168 C4V6RF 9998996 IC50 > 5000 nM T72168 CC4WY6 10024990 IC50 = 1000 nM T72168 CSM0W3 10026120 IC50 > 2000 nM T72168 CFY67M 10070808 IC50 = 2219 nM T72168 C9T4HR 10071810 IC50 = 1100 nM T72168 CQ3LD1 10091351 IC50 = 1600 nM T72168 C16HAK 10094808 IC50 > 2000 nM T72168 CR0DX5 10126475 IC50 > 1130 nM T72168 CHS18G 10126476 IC50 > 2000 nM T72168 CR0BP6 10126871 IC50 = 380 nM T72168 CV5PQ0 10126940 IC50 = 500 nM T72168 CVF40M 10127159 IC50 = 350 nM T72168 C3CRZ1 10127269 IC50 = 450 nM T72168 CPB60D 10127340 IC50 = 760 nM T72168 CKMW98 10128037 IC50 = 585 nM T72168 C1GI3D 10150743 IC50 = 220 nM T72168 CZKF71 10150825 IC50 = 400 nM T72168 CYR0U5 10150851 IC50 > 2000 nM T72168 CVO1F7 10151165 IC50 = 405 nM T72168 C6EC1P 10151186 IC50 = 405 nM T72168 CQ14RM 10151357 IC50 = 535 nM T72168 CW4Y2K 10151995 IC50 = 1650 nM T72168 C0MX7K 10157532 IC50 = 893 nM T72168 CL0U4N 10172897 IC50 = 400 nM T72168 CG0VH8 10173354 IC50 = 1250 nM T72168 CU6D8W 10173525 IC50 = 170 nM T72168 C8L7HJ 10179031 IC50 = 683 nM T72168 C41YRZ 10194268 IC50 > 740 nM T72168 CX4F7Z 10194607 IC50 > 2000 nM T72168 CV0LE4 10194889 IC50 > 1000 nM T72168 C3O7WH 10215978 IC50 = 1350 nM T72168 C1SG4N 10216152 IC50 > 1420 nM T72168 CD0YT7 10216465 IC50 = 940 nM T72168 C1FGX9 10216535 IC50 = 415 nM T72168 CW7QX2 10216536 IC50 = 720 nM T72168 CG9OH4 10216697 IC50 = 1050 nM T72168 CXN4W1 10216788 IC50 = 1100 nM T72168 CUGN98 10217411 IC50 = 910 nM T72168 CJ9BE0 10222329 IC50 = 651 nM T72168 C84SRT 10223610 IC50 = 2154 nM T72168 CUYO17 10237223 IC50 > 1300 nM T72168 CWYK62 10238100 IC50 = 435 nM T72168 C1R8GY 10238297 IC50 = 900 nM T72168 CNB1V3 10238624 IC50 = 190 nM T72168 CPGF94 10238831 IC50 > 2000 nM T72168 C2AZH1 10238961 IC50 = 175 nM T72168 CSA4R3 10252455 IC50 > 2000 nM T72168 C7EGH2 10252527 IC50 = 120 nM T72168 CR59SC 10271193 IC50 = 22897 nM T72168 CPIS57 10271557 IC50 = 2252 nM T72168 CUQC81 10287415 IC50 > 1000 nM T72168 C5RC7X 10287444 IC50 = 510 nM T72168 CJT2G8 10287863 IC50 = 1400 nM T72168 C1M6WY 10288006 IC50 = 320 nM T72168 CO6UP3 10288155 IC50 = 875 nM T72168 C6C2IK 10288565 IC50 = 195 nM T72168 CNEO49 10289020 IC50 = 104 nM T72168 CLJU03 10298892 Ki = 3914 nM T72168 C9UYG8 10309447 IC50 > 1050 nM T72168 C8FM2D 10309755 IC50 = 1800 nM T72168 C1OV7M 10309756 IC50 = 715 nM T72168 C9TI4A 10310063 IC50 = 1035 nM T72168 CP9AE0 10310476 IC50 > 512 nM T72168 CV52EN 10310809 IC50 = 140 nM T72168 CR1L5N 10311251 IC50 = 104 nM T72168 CX7WS4 10316069 IC50 = 354 nM T72168 CQP1Y7 10340204 IC50 = 1525 nM T72168 CEJ78I 10365592 IC50 > 2000 nM T72168 CDBZ06 10372181 IC50 = 120 nM T72168 C14AIB 10384345 IC50 = 970 nM T72168 CZ5CJ3 10423330 IC50 > 10000 nM T72168 C5I3BG 10428464 Ki = 12 nM T72168 C1KE6C 10446402 IC50 = 2050 nM T72168 C0NT9D 10454007 IC50 > 5000 nM T72168 C85RBN 10474264 IC50 > 2000 nM T72168 CUL8O4 10475384 IC50 > 5000 nM T72168 CPX65M 10477088 IC50 = 130 nM T72168 C5AP6C 10503520 IC50 > 10000 nM T72168 CBEC38 10596252 IC50 = 1000 nM T72168 CC8T7J 10598305 IC50 = 1062 nM T72168 CO3V0S 10622594 IC50 = 977 nM T72168 C02ZMG 10643956 IC50 = 748 nM T72168 CYNG45 10668755 IC50 > 10000 nM T72168 CYRQ10 10691647 Ki = 1100 nM T72168 CVD2Y9 10717098 IC50 > 10000 nM T72168 CAT1X8 10741366 IC50 = 1068 nM T72168 CB3JD0 10763832 IC50 = 1358 nM T72168 C07BOR 10787258 IC50 = 2035 nM T72168 C1CRQ5 10811045 IC50 > 10000 nM T72168 CN1H5Z 10832792 IC50 = 1592 nM T72168 CHU9A4 10873317 IC50 = 334 nM T72168 CHU10G 10960295 IC50 = 1850 nM T72168 C6LYG7 11090322 IC50 > 1000 nM T72168 CXS6J7 11155441 Ki = 10 nM T72168 CQUV78 11176984 IC50 = 23 nM T72168 CL97OU 11212803 IC50 = 540 nM T72168 C4U0DF 11213029 Ki = 980 nM T72168 CRN4V2 11232136 IC50 > 3000 nM T72168 C8XPZ4 11269445 IC50 > 2000 nM T72168 C4HNB8 11269886 IC50 = 1050 nM T72168 CC0XI4 11279959 IC50 = 440 nM T72168 C4SC0W 11281576 IC50 > 5000 nM T72168 C8YL6K 11282486 IC50 = 1700 nM T72168 CUX0S2 11282904 Ki = 21 nM T72168 CIY9H5 11291999 IC50 = 1800 nM T72168 C0IQ9K 11304445 IC50 = 160 nM T72168 C0XUF2 11305564 IC50 > 5000 nM T72168 CXC9G3 11327341 IC50 > 2000 nM T72168 CT9Y4O 11339440 IC50 = 2300 nM T72168 C8FQ9B 11375180 IC50 = 21000 nM T72168 CP2DL0 11377050 IC50 = 1000 nM T72168 C76VYN 11382721 IC50 > 2000 nM T72168 CV4RO2 11384310 IC50 = 48 nM T72168 CXW40M 11384346 IC50 > 2000 nM T72168 CU7IE0 11410199 IC50 = 690 nM T72168 CO20QH 11416730 IC50 = 155 nM T72168 C5WO0U 11429662 IC50 > 5000 nM T72168 CD2Q3F 11474917 IC50 = 83 nM T72168 CC75NQ 11477616 Ki = 430 nM T72168 CQ62KS 11485693 IC50 > 3000 nM T72168 C9Q1NY 11494167 Ki = 32 nM T72168 CFLQ08 11495227 IC50 = 320 nM T72168 C03NYX 11495549 IC50 = 90 nM T72168 CR40IH 11516847 IC50 = 1800 nM T72168 CP4F8X 11517412 IC50 = 280 nM T72168 C2PB6Z 11530605 Ki = 930 nM T72168 C1R6DC 11531942 IC50 = 140 nM T72168 CZ1HA3 11538472 IC50 = 615 nM T72168 CFC1Z4 11538799 IC50 = 1100 nM T72168 CBK60G 11559947 IC50 > 2000 nM T72168 C1D9YS 11560003 IC50 > 2000 nM T72168 CB37YF 11566981 Ki = 145 nM T72168 C8WJ2F 11567609 IC50 = 780 nM T72168 C0SCT6 11588584 IC50 = 810 nM T72168 C3MW1D 11589982 IC50 = 220 nM T72168 C03QYZ 11590471 IC50 = 110 nM T72168 CAO2P1 11596392 IC50 > 2000 nM T72168 CSB97O 11617028 Ki = 21 nM T72168 CRL3A7 11632925 IC50 = 120 nM T72168 CQB0E3 11633482 IC50 = 65 nM T72168 C9DNG1 11640164 IC50 = 580 nM T72168 C1RJ3I 11646689 IC50 = 1000 nM T72168 CX3L5S 11647533 IC50 = 80 nM T72168 C4S5RG 11655053 IC50 = 175 nM T72168 CDOZ32 11661172 IC50 = 590 nM T72168 C0LEZ3 11667800 Ki = 890 nM T72168 C5XEN0 11668719 IC50 = 220 nM T72168 CZPK72 11682989 IC50 = 80 nM T72168 CCK83U 11690269 IC50 = 160 nM T72168 CY07JH 11696378 IC50 > 2000 nM T72168 CBU02W 11696959 IC50 = 640 nM T72168 C2S9IT 11697271 IC50 = 1900 nM T72168 CGR32I 11697882 IC50 = 340 nM T72168 C75IBX 11704529 IC50 = 90 nM T72168 CGX54N 11704756 IC50 = 210 nM T72168 CO2N1W 11710364 IC50 = 1550 nM T72168 CZ52YQ 11710766 IC50 < 500 nM T72168 C8OPA1 11710962 IC50 = 855 nM T72168 CW3N8H 11711766 IC50 = 280 nM T72168 COEU05 11719039 IC50 = 100 nM T72168 CZ0B7H 11731863 IC50 = 1900 nM T72168 CQO76Z 11741168 IC50 > 2000 nM T72168 C87YNC 11741891 IC50 = 150 nM T72168 CH92VI 11743259 IC50 = 310 nM T72168 C5HLU8 11750204 IC50 = 380 nM T72168 CY1F4I 11752649 Ki = 670 nM T72168 CQU0E7 11774868 IC50 = 435 nM T72168 C4U8KY 12085089 IC50 = 162 nM T72168 C14LTD 15463551 IC50 > 1000 nM T72168 C3QOV0 16099227 IC50 = 430 nM T72168 CW6LO1 16099229 IC50 > 2000 nM T72168 C2R4PK 16099231 IC50 = 450 nM T72168 C9KM7X 16099232 IC50 = 1900 nM T72168 C05CYN 16099234 IC50 = 1600 nM T72168 CJQ8A1 16099236 IC50 = 450 nM T72168 CA72YW 16099237 IC50 > 2000 nM T72168 CS07DB 16099238 IC50 = 98 nM T72168 C42ESN 16099240 IC50 = 580 nM T72168 CMZ91J 16099242 IC50 > 2000 nM T72168 CF69RC 16099243 IC50 > 2000 nM T72168 C60GEM 16099245 IC50 = 1500 nM T72168 CE48CS 16099246 IC50 = 620 nM T72168 CTF2M7 16099247 IC50 = 130 nM T72168 CX9BK2 16099248 IC50 = 775 nM T72168 CN6PA9 16099249 IC50 = 350 nM T72168 C9Z6AK 16099250 IC50 = 120 nM T72168 C5Z8HR 16099251 IC50 = 91 nM T72168 CWK76M 16099252 IC50 = 880 nM T72168 C3BU9M 16216822 IC50 = 290 nM T72168 C1Q5SV 16220168 IC50 = 510 nM T72168 CH6CN0 16658901 Ki > 10000 nM T72168 CU9LS2 16661702 EC50 = 5000 nM T72168 C1UY8J 16666386 IC50 > 1000 nM T72168 CWK35C 16730429 IC50 = 8700 nM T72168 CSKX58 17758233 Ki = 410 nM T72168 C7CPW9 17758234 Ki = 48 nM T72168 CI5KT6 17758236 Ki = 42 nM T72168 C3FP7L 17921933 IC50 = 3162 nM T72168 CX03YG 18188955 IC50 = 1220 nM T72168 CR19ST 18512166 IC50 = 310 nM T72168 CEN14G 18512334 IC50 = 4000 nM T72168 CS9CI5 18551230 IC50 = 30 nM T72168 CBI64N 18551237 IC50 = 130 nM T72168 C5ZYJ0 20231824 Ki = 952 nM T72168 CEH7V5 20786216 IC50 > 1000 nM T72168 C97WCO 21941658 IC50 = 1.259 nM T72168 CCI89R 21948853 IC50 > 1000 nM T72168 CB2SF4 21948904 IC50 > 1000 nM T72168 C2ZP7V 22218142 IC50 = 1500 nM T72168 C1QTK4 22398492 IC50 = 240 nM T72168 C6CSB4 22398502 IC50 > 2000 nM T72168 CR8N1E 22398506 IC50 = 1420 nM T72168 CM83TU 22398533 IC50 = 265 nM T72168 C34LHW 22398559 IC50 = 910 nM T72168 CJBW90 22398592 IC50 > 2000 nM T72168 CEJ65O 22398627 IC50 = 415 nM T72168 CZI4C6 24739672 Ki = 1000 nM T72168 CS23KY 24739834 Ki = 1390 nM T72168 C1M9QG 24739836 Ki = 1770 nM T72168 CG5SJ0 24739997 Ki = 1490 nM T72168 C7Z1HW 24740156 Ki = 1440 nM T72168 CTE1N2 24748569 EC50 > 10000 nM T72168 C4WYE7 24749678 Ki = 1.56 nM T72168 CY2JS4 24749684 Ki = 1.51 nM T72168 C2QHO3 24749808 Ki = 0.319 nM T72168 C5S6JN 24780149 IC50 > 1000 nM T72168 CW5TJ7 24781731 IC50 > 1000 nM T72168 C1JTW2 24851053 Ki = 0.342 nM T72168 CC53XL 24860583 Ki > 3000 nM T72168 C58RHY 24883011 IC50 = 80 nM T72168 CW35CK 24883012 IC50 = 41 nM T72168 C3SC0V 24883054 IC50 = 76 nM T72168 C4SA6C 24883055 IC50 = 15 nM T72168 C5LZK2 24895096 IC50 = 1350 nM T72168 COGP96 24936313 IC50 > 5000 nM T72168 CVY09S 24936449 IC50 > 5000 nM T72168 C06PDG 24952192 EC50 > 5000 nM T72168 CG1CF9 24952193 EC50 > 5000 nM T72168 CZC7L8 24953162 IC50 > 10000 nM T72168 C4W7BN 24954947 IC50 > 10000 nM T72168 C6XC2R 24954951 IC50 > 20000 nM T72168 CYES17 24957737 Ki > 3000 nM T72168 C83YKB 24961057 Ki > 1000 nM T72168 CIGM27 24983460 IC50 = 280 nM T72168 CHY0D7 25013322 IC50 > 10000 nM T72168 C0TPS5 25013653 IC50 > 10000 nM T72168 CWU91M 25013811 IC50 > 10000 nM T72168 CSH29L 25013812 IC50 > 10000 nM T72168 C7QCX0 25052023 IC50 = 2.4 nM T72168 CAW8M0 25070694 IC50 = 2800 nM T72168 C21XDY 25145083 Ki > 10000 nM T72168 CS6JQ1 25167502 Ki = 155 nM T72168 C0XPW9 25168896 IC50 = 340 nM T72168 CUL27D 25168900 IC50 = 260 nM T72168 CEV2D7 25205475 IC50 = 260 nM T72168 C9S0ZW 25205477 IC50 = 330 nM T72168 C49KHR 25206116 IC50 = 510 nM T72168 C9FM2U 42642501 Ki <= 10 nM T72168 CXZ35T 44193145 Ki = 656 nM T72168 C2MOF7 44193146 Ki = 378 nM T72168 CWR6X1 44193147 Ki = 2250 nM T72168 C3JOW4 44193245 Ki = 1470 nM T72168 CHGI03 44251606 IC50 = 475 nM T72168 C0OA6M 44264483 IC50 > 10000 nM T72168 COCE32 44264569 IC50 > 10000 nM T72168 CI0TN2 44264577 IC50 > 10000 nM T72168 CXOR54 44264579 IC50 > 10000 nM T72168 C01HSQ 44264588 IC50 > 10000 nM T72168 CDB54J 44305270 IC50 > 1000 nM T72168 C0XLN6 44305556 IC50 > 1000 nM T72168 C1UK4M 44305720 IC50 = 1889 nM T72168 CH4PU5 44305819 IC50 = 2484 nM T72168 C6N1AR 44305929 IC50 2871 nM T72168 C73CXK 44354006 IC50 = 363 nM T72168 C0N3TD 44354884 IC50 = 2700 nM T72168 CPQ2A6 44354885 IC50 = 1000 nM T72168 CM0G1V 44354886 IC50 = 2000 nM T72168 CL6G3Q 44355066 IC50 = 2100 nM T72168 CSAU31 44377064 IC50 > 10000 nM T72168 C7H9NC 44377081 IC50 > 10000 nM T72168 C60DYH 44377090 IC50 = 2000 nM T72168 CVH2R3 44377098 IC50 = 2900 nM T72168 CYLI63 44377110 IC50 > 10000 nM T72168 CQX39I 44377356 IC50 = 570 nM T72168 C9FJW4 44377382 IC50 = 1900 nM T72168 C13SYV 44396250 Ki = 300 nM T72168 CB1P0S 44396251 Ki = 80 nM T72168 CHY1C3 44396271 Ki = 590 nM T72168 C29MBI 44396272 Ki = 310 nM T72168 C4TQ6N 44396282 Ki = 440 nM T72168 CH2Y3L 44396283 Ki = 190 nM T72168 CWZB52 44396284 Ki = 850 nM T72168 CD80LM 44396296 Ki > 1000 nM T72168 C6SI5L 44396297 Ki > 1000 nM T72168 CR4H1E 44396316 Ki = 510 nM T72168 C45LRH 44396317 Ki = 140 nM T72168 C5JG6H 44396330 Ki > 1000 nM T72168 CA8V4G 44396331 Ki > 1000 nM T72168 C57CPQ 44396332 Ki = 310 nM T72168 CXHF58 44403036 IC50 = 215 nM T72168 C6JNI4 44403038 IC50 = 60 nM T72168 C45SOW 44403039 IC50 = 315 nM T72168 CXZ4S3 44426781 Ki = 3490 nM T72168 C8HO4K 44426782 Ki = 585 nM T72168 C0FEN3 44426790 Ki = 298 nM T72168 C19MJP 44426793 Ki = 527 nM T72168 C1ZDA4 44426795 Ki = 1270 nM T72168 CIOW01 44431179 IC50 = 520 nM T72168 C3SJ5V 44433504 Ki = 7.5 nM T72168 C2SCP7 44435606 IC50 = 1600 nM T72168 CH5E3L 44435611 IC50 > 1300 nM T72168 CDO62N 44435656 IC50 = 650 nM T72168 C9TP4C 44435662 IC50 = 345 nM T72168 C19TMW 44435663 IC50 = 730 nM T72168 C90WUC 44435667 IC50 = 430 nM T72168 CHFB89 44435668 IC50 = 300 nM T72168 C8IWK2 44435669 IC50 = 250 nM T72168 CYG7X4 44473146 IC50 > 10000 nM T72168 CR5SI0 44476535 EC50 > 10000 nM T72168 CM29JD 44516036 IC50 > 10000 nM T72168 CR19IH 44543858 IC50 > 2000 nM T72168 C05HEP 44543860 IC50 > 2000 nM T72168 C45ZHO 44543969 IC50 > 2000 nM T72168 C25OXZ 44544094 IC50 > 2000 nM T72168 C7JIF6 44544321 IC50 > 2000 nM T72168 CF6V4G 44563171 EC50 > 10000 nM T72168 C8BGL6 44585565 IC50 > 3000 nM T72168 CIJP09 44605898 IC50 > 10000000 nM T72168 C9PLK4 45263610 IC50 > 2000 nM T72168 C78JKD 45265930 IC50 = 1100 nM T72168 C08UBE 45272032 IC50 > 10000 nM T72168 C57EZH 45275745 IC50 = 110 nM T72168 CU7D0O 45278780 IC50 = 3.7 nM T72168 CY8A1D 45278857 IC50 = 3.1 nM T72168 CGX87F 45279098 IC50 = 6.5 nM T72168 CL9P2A 45380783 IC50 = 3.8 nM T72168 CKC0B7 46237842 IC50 = 59 nM T72168 C4KN0J 46237981 IC50 = 31 nM T72168 C7KW8T 46883839 EC50 > 10000 nM T72168 CZSG25 46883893 EC50 > 10000 nM T72168 C72MUY 46889765 IC50 > 5000 nM T72168 C6DVO1 46889848 IC50 > 10000 nM T72168 CZ90FC 46894119 Ki = 9 nM T72168 C04KWS 46913888 IC50 = 54 nM T72168 C1U7QL 46913889 IC50 = 52 nM T72168 C3Q7RI 46913890 IC50 = 6 nM T72168 CY7D0I 46913891 IC50 = 80 nM T72168 CQ93ML 46913892 IC50 = 135 nM T72168 C1ZRD2 46914168 IC50 = 1620 nM T72168 CWV42M 46914169 IC50 = 3740 nM T72168 CK6SJ3 46914453 IC50 = 275 nM T72168 C4HQ5Y 46914584 IC50 = 223 nM T72168 C9F4PR 46914585 IC50 = 4340 nM T72168 CZE49A 46914586 IC50 = 553 nM T72168 CGS9U8 46914587 IC50 = 41 nM T72168 C34EDY 46914588 IC50 = 21 nM T72168 CLCI21 46914734 IC50 = 13 nM T72168 C2NM6E 46914737 IC50 = 25 nM T72168 CKP01L 46914738 IC50 = 58 nM T72168 CP91XE 46914741 IC50 = 89 nM T72168 C3Q5PE 46914742 IC50 = 4 nM T72168 C6OG0A 46914743 IC50 = 7 nM T72168 C1TMA8 46914744 IC50 = 150 nM T72168 CE7KZ8 46914881 IC50 = 83 nM T72168 CI0Y4F 46914882 IC50 > 10000 nM T72168 C8HWO7 46914883 IC50 = 784 nM T72168 C6FN4G 46914884 IC50 = 246 nM T72168 CXY74T 46914885 IC50 = 9730 nM T72168 CF1D5Q 46914886 IC50 = 488 nM T72168 CVGF35 46914887 IC50 > 500 nM T72168 C4ZPR6 46915029 IC50 = 180 nM T72168 CXR29C 46915030 IC50 > 10000 nM T72168 C9NC0K 46915031 IC50 = 1440 nM T72168 CY3O2C 46915043 IC50 = 41 nM T72168 CHG94E 46915044 IC50 = 32 nM T72168 CK85FJ 46915045 IC50 = 101 nM T72168 CQ6J3N 46915201 IC50 = 2080 nM T72168 CC84WO 46915202 IC50 = 8360 nM T72168 CTM2J5 46915203 IC50 = 31 nM T72168 C75IFZ 46915353 IC50 = 16 nM T72168 CJW51A 46915354 IC50 = 26 nM T72168 CX70GY 46915355 IC50 = 15.2 nM T72168 CPTL45 46915356 IC50 = 2 nM T72168 C39SUV 46915640 IC50 = 243 nM T72168 CX6WK5 46915641 IC50 = 535 nM T72168 CW8J2E 46915642 IC50 = 56 nM T72168 C05YTF 46915643 IC50 = 284 nM T72168 CMW7E4 46915644 IC50 = 56 nM T72168 CA43UG 46915645 IC50 > 127 nM T72168 CJ3DN2 46915781 IC50 > 1000 nM T72168 C4L1JF 46915782 IC50 = 383 nM T72168 CB4X3D 46915783 IC50 > 10000 nM T72168 CK7DI0 46915784 IC50 > 10000 nM T72168 CU7L4T 46915785 IC50 = 10000 nM T72168 CE9OU3 46915786 IC50 = 410 nM T72168 CI3E2M 46915787 IC50 = 763 nM T72168 C1BV5K 46916070 IC50 = 3650 nM T72168 C06JHQ 46916071 IC50 = 441 nM T72168 CQ37UY 46916072 IC50 = 1590 nM T72168 C38HIP 46916073 IC50 = 1290 nM T72168 CPK95L 46916074 IC50 = 151 nM T72168 C7NC4B 46917090 IC50 = 2.8 nM T72168 C2LCJ7 46937290 IC50 = 210 nM T72168 CKQ8J3 46937431 IC50 > 2000 nM T72168 CL7P3N 46938234 IC50 = 1.8 nM T72168 COS28G 46938235 IC50 = 18 nM T72168 CFJT93 46938236 IC50 = 7.6 nM T72168 CHL70M 46938239 IC50 = 4.1 nM T72168 C8P7JH 46938914 IC50 > 2000 nM T72168 CY95VK 46938915 IC50 > 2000 nM T72168 CVX25Q 46938916 IC50 = 220 nM T72168 C2V5AT 46939019 IC50 = 480 nM T72168 C5R6GI 46939020 IC50 = 390 nM T72168 CF1BX0 46939115 IC50 > 2000 nM T72168 C4P0EU 46939116 IC50 = 160 nM T72168 CD6B7X 46939395 IC50 = 58 nM T72168 C1KXF2 46939396 IC50 > 2000 nM T72168 CVN4W1 47958757 IC50 = 168 nM T72168 CX0NO8 49782554 EC50 < 15848.93 nM T72168 CC7T8Q 49782555 EC50 < 15848.93 nM T72168 CD07EV 49782777 EC50 < 15848.93 nM T72168 C43UKW 49782778 IC50 < 14421.15 nM T72168 C2JTF0 49782779 EC50 < 15848.93 nM T72168 CS7KX9 49782780 IC50 < 12560.3 nM T72168 C36RYU 49782781 IC50 = 5140.44 nM T72168 C8OA0C 49782985 EC50 < 15848.93 nM T72168 C5Y6QU 49782986 EC50 < 15848.93 nM T72168 CB8V7R 49782987 EC50 < 15848.93 nM T72168 CU3S6H 49836028 EC50 > 5000 nM T72168 C96SLW 49851364 EC50 > 5000 nM T72168 CDN4K6 49851369 EC50 > 5000 nM T72168 C4YXN1 49851467 EC50 > 5000 nM T72168 CUD91T 49862248 EC50 > 10000 nM T72168 C5NX4D 49864061 IC50 = 2530 nM T72168 CPH9D8 49864098 IC50 = 69 nM T72168 CMS1N3 49864127 IC50 = 15 nM T72168 CTE0N7 49864128 IC50 = 720 nM T72168 COP7W2 49864129 IC50 = 127 nM T72168 CCKJ45 49864153 IC50 = 849 nM T72168 C19FRV 49864154 IC50 = 65 nM T72168 CWGD27 49864174 IC50 = 146 nM T72168 C9YCN1 49864175 IC50 = 39 nM T72168 CTKV39 49864176 IC50 = 26 nM T72168 CZ8J1V 50942115 Ki = 800 nM T72168 C23OEF 50942312 EC50 > 10000 nM T72168 CX1KO8 51346768 Ki = 849 nM T72168 C7N9TD 51346823 Ki = 1518 nM T72168 C0WDX3 51347001 Ki = 1115 nM T72168 CF8DK7 51347002 Ki = 3170 nM T72168 CTH45Q 52918523 IC50 > 10000 nM T72168 CL8D1Z 52921432 IC50 = 130 nM T72168 CEC4I7 52941608 IC50 = 230 nM T72168 CDV90J 52942528 IC50 > 1000 nM T72168 C8Y9SU 52944898 IC50 > 1000 nM T72168 CK5UT4 53317489 Ki = 126 nM T72168 CM0LU1 53318659 Ki = 1200 nM T72168 CUD48O 53320087 Ki = 0.64 nM T72168 CD0N1K 53323476 IC50 = 356 nM T72168 CYH3V0 53325642 Ki = 86.8 nM T72168 C82DYI 53326614 Ki > 4170 nM T72168 CJCP75 53359074 EC50 > 5000 nM T72168 C9H5YE 53361128 EC50 > 5000 nM T72168 CUR24K 53875787 IC50 = 2800 nM T72168 C1JR5W 54576068 IC50 = 24 nM T72168 CS62XZ 54590901 IC50 = 53.9 nM T72168 C30XLO 54592009 Ki = 6.3 nM T72168 CCS8R6 54592010 IC50 = 39 nM T72168 CML2E7 54592011 IC50 = 86 nM T72168 CRVB01 54592087 IC50 = 266 nM T72168 C7W1BA 54592088 IC50 = 109 nM T72168 C9N3IS 54592089 IC50 = 56 nM T72168 C2GML6 54592090 IC50 = 33 nM T72168 C05FVP 54592092 IC50 = 19 nM T72168 C9W5DZ 56593984 EC50 > 5000 nM T72168 CF3G2M 56925477 IC50 = 36 nM T72168 CZ7O8G 56925478 IC50 = 69 nM T72168 CV5C0T 56925479 IC50 > 10000 nM T72168 C9ITY0 56925480 IC50 > 10000 nM T72168 C3M4TE 56925570 IC50 = 920 nM T72168 CZ4I2J 56925571 IC50 = 6800 nM T72168 CW87RG 56925573 IC50 = 2000 nM T72168 C4Z5LF 56925574 IC50 = 4100 nM T72168 CKF8Z3 56925575 IC50 = 1300 nM T72168 CY20OR 56925668 IC50 > 10000 nM T72168 C30DAL 56925669 IC50 = 600 nM T72168 CQHA65 56925670 IC50 = 310 nM T72168 CJP31U 56925671 IC50 = 270 nM T72168 CV86DS 56925673 IC50 = 2700 nM T72168 CI3S6F 56925790 IC50 = 5300 nM T72168 CTY1Q9 56925791 IC50 = 1100 nM T72168 CH40YG 56925792 IC50 = 960 nM T72168 C2PLD4 56925793 IC50 = 260 nM T72168 CU02HT 56925794 IC50 = 570 nM T72168 CM19WI 56925904 IC50 > 10000 nM T72168 CA7BX4 56925905 IC50 = 440 nM T72168 CTR7X3 56925906 IC50 = 1100 nM T72168 C39VBK 56925907 IC50 = 430 nM T72168 CV7EN5 56925908 IC50 = 320 nM T72168 CU69SK 56925909 IC50 = 590 nM T72168 CAMI87 56925910 IC50 = 700 nM T72168 CTG9I7 56926011 IC50 = 70 nM T72168 CPD82H 56968080 IC50 = 7.1 nM T72168 CM0SG2 57390990 IC50 = 1100 nM T72168 CU8AN3 57392780 IC50 = 790 nM T72168 CX12JM 57392781 IC50 = 45 nM T72168 C9OMW1 57392782 IC50 = 405 nM T72168 C30JOV 57394501 IC50 = 190 nM T72168 CINU04 57396254 IC50 = 225 nM T72168 C1O6JU 57396255 IC50 = 230 nM T72168 CVOB64 57399718 IC50 = 610 nM T72168 CF83VM 57401459 EC50 > 5000 nM T72168 C7W3YD 57401479 IC50 = 430 nM T72168 CR6L7E 57403222 IC50 = 1450 nM T72168 CPU6W7 57473898 IC50 = 80 nM T72168 CEJ25K 57473899 IC50 = 270 nM T72168 CUJ08D 57474008 IC50 = 70 nM T72168 CDB0F1 57503322 IC50 = 39 nM T72168 CIDS61 57503325 IC50 = 19 nM T72168 C2U1GQ 57524309 IC50 = 22 nM T72168 C0BDS9 57585514 IC50 < 2 nM T72168 CM17UZ 57585515 IC50 = 47 nM T72168 CYGU85 57585534 IC50 = 1.3 nM T72168 C3WG0L 57666312 Ki = 1100 nM T72168 C43GDR 57666397 Ki = 290 nM T72168 CTM6K5 57690900 IC50 > 5000 nM T72168 CB2I7A 57748722 Ki <= 10 nM T72168 CT9Y6X 57748723 Ki <= 10 nM T72168 C6J0HD 57748748 Ki <= 10 nM T72168 C2MFH6 57748755 Ki <= 10 nM T72168 CMR56T 57748765 Ki <= 10 nM T72168 C05UIP 57748768 Ki <= 10 nM T72168 CH2PV6 57748780 Ki = 0.79 nM T72168 CL13HZ 57748781 Ki = 0.4 nM T72168 C7UH3N 57748789 Ki <= 10 nM T72168 C2YT7S 57748790 Ki = 0.23 nM T72168 C1KZT3 57906156 IC50 = 500 nM T72168 C3IN9F 57983276 IC50 = 170 nM T72168 CJ6Y1B 58026134 IC50 > 2000 nM T72168 C19XQV 58026164 IC50 > 2000 nM T72168 CR7H3O 58026170 IC50 > 2000 nM T72168 C7XL3D 58026176 IC50 > 2000 nM T72168 CT1EM3 58064710 IC50 = 3.7 nM T72168 C8S3EQ 58064714 IC50 = 2.7 nM T72168 CPI62D 58064720 IC50 = 2.2 nM T72168 CL42XF 58064726 IC50 = 4.3 nM T72168 CPL9A6 58064729 IC50 = 55.9 nM T72168 CRFS78 58064730 IC50 = 3.3 nM T72168 CN1J3V 58064734 IC50 = 17.8 nM T72168 CA0SH5 58064735 IC50 = 4.4 nM T72168 CI7BP4 58064741 IC50 = 21.4 nM T72168 C2FZA7 58064756 IC50 = 9.4 nM T72168 C3AMO0 58064757 IC50 = 4450 nM T72168 C47AUR 58392644 EC50 = 2.5 nM T72168 C9CQS0 58392665 EC50 = 3.2 nM T72168 CXF39M 58392685 EC50 > 3000 nM T72168 C7FXH3 58392721 EC50 > 3000 nM T72168 CJDN90 58392790 EC50 = 1.6 nM T72168 CO59DQ 58392803 EC50 > 3000 nM T72168 C5K9PJ 58483018 IC50 = 1.2 nM T72168 C4C2FT 58599563 IC50 = 1300 nM T72168 CWAD17 58731166 Ki <= 500 nM T72168 CNE02T 58731180 Ki <= 500 nM T72168 CVS58C 58731199 Ki <= 500 nM T72168 C3VU0Q 58731202 Ki <= 500 nM T72168 C03HFM 58731234 Ki <= 500 nM T72168 CADQ18 58731243 Ki <= 500 nM T72168 CI7XQ5 58731245 Ki <= 500 nM T72168 C67UET 58731323 Ki <= 500 nM T72168 C0JL7A 58973277 IC50 > 1000 nM T72168 CY38HG 59233337 Ki > 1000 nM T72168 CUX4E7 59233347 Ki > 3333 nM T72168 CO63VJ 59233364 Ki > 1000 nM T72168 C2A9JO 59251119 IC50 > 5000 nM T72168 CD8A6P 59281281 IC50 = 49 nM T72168 CBZ0M5 59281312 IC50 = 170 nM T72168 CCT59B 59281329 IC50 = 510 nM T72168 CQI5C4 59281343 IC50 = 38 nM T72168 CH5E1F 59281346 IC50 > 10000 nM T72168 CPE83R 59281354 IC50 = 180 nM T72168 CI9EP1 59281363 IC50 = 8.4 nM T72168 CQ2BO1 59281403 IC50 = 51 nM T72168 CP78RD 59281411 IC50 = 95 nM T72168 CCNU12 59281412 IC50 = 10 nM T72168 C7HVB1 59281416 IC50 = 490 nM T72168 CE5A0V 59281447 IC50 = 75 nM T72168 CZT9S6 59281449 IC50 = 430 nM T72168 CIKQ89 59281508 IC50 = 990 nM T72168 CE1A7J 59281531 IC50 = 680 nM T72168 CK9JZ4 59281538 IC50 = 36 nM T72168 C4TG5U 59281540 IC50 = 22 nM T72168 CPC80S 59281541 IC50 = 64 nM T72168 CXS5C4 59281543 IC50 = 250 nM T72168 C7KPR9 59281566 IC50 = 150 nM T72168 CUJP64 59281599 IC50 = 600 nM T72168 CYZI85 59556974 IC50 > 10000 nM T72168 C5C3AO 59770003 Ki = 2.48 nM T72168 CH36PL 59807625 IC50 < 500 nM T72168 C54ATL 59807726 IC50 < 500 nM T72168 C8S7OB 59808080 IC50 < 500 nM T72168 CYU57B 59808129 IC50 < 500 nM T72168 C2TNO8 60026286 IC50 > 2000 nM T72168 CZE5J8 60026377 IC50 > 2000 nM T72168 C0LDS2 60026592 IC50 = 1150 nM T72168 C31PTC 60026641 IC50 > 2000 nM T72168 C67NSE 60026675 IC50 > 2000 nM T72168 C6GP5R 60026731 IC50 = 720 nM T72168 C5M8HV 60026772 IC50 = 1200 nM T72168 CI36XS 60026787 IC50 > 2000 nM T72168 C3JD8M 60026802 IC50 > 2000 nM T72168 CE9MI4 60026817 IC50 = 1900 nM T72168 C04EKW 60026878 IC50 > 2000 nM T72168 CPRW14 66991384 IC50 = 160 nM T72168 CYP31Z 66995780 IC50 = 3050 nM T72168 CK36QI 66996020 IC50 > 10000 nM T72168 CJ09TZ 66996063 IC50 = 2225 nM T72168 C3EU7N 66996137 IC50 = 276 nM T72168 C1CXY9 66996546 IC50 = 401 nM T72168 C9Y2DN 66996560 IC50 = 727 nM T72168 C9LOZ1 66996568 IC50 = 1181 nM T72168 CH39DP 67053383 IC50 > 2000 nM T72168 C3LF8O 67053425 IC50 > 2000 nM T72168 CMYP75 67415874 IC50 = 100 nM T72168 CQU8E3 68031408 IC50 = 11 nM T72168 C1FK3D 69081573 IC50 = 31 nM T72168 CB6HX8 69082589 IC50 = 480 nM T72168 C43PON 69675755 IC50 = 9.4 nM T72168 COR52G 69675880 IC50 = 13 nM T72168 C9Q7VH 70561849 IC50 = 39 nM T72168 CARO49 70685018 Ki = 150 nM T72168 C5QPC0 70697572 Ki = 170 nM T72168 C94FCP 71452686 IC50 = 3000 nM T72168 CF08ME 71457470 Ki = 0.4 nM T72168 CEO5G4 71461616 IC50 = 1900 nM T72168 C78IOK 71467161 IC50 = 310 nM T72168 C1MHC0 71467246 IC50 = 47 nM T72168 C4B0IC 71467248 IC50 = 26 nM T72168 CYW34A 71519686 IC50 = 120 nM T72168 CGK4S8 71543393 Ki = 1450 nM T72168 C83YJF 71544946 IC50 = 39 nM T72168 CK2O1Z 71545110 IC50 = 54 nM T72168 C0LD8K 71548690 IC50 = 270 nM T72168 C19CGP 71548691 IC50 = 1700 nM T72168 C4BE6G 71548692 IC50 = 1110 nM T72168 CCK7Q3 71548693 IC50 = 240 nM T72168 CK9S0J 71548694 IC50 = 1440 nM T72168 CT9Y5D 71549558 Ki = 2 nM T72168 C8ZX0F 71549573 IC50 = 180 nM T72168 COQ5C4 71549690 IC50 = 230 nM T72168 CE7NZ0 71549691 IC50 = 190 nM T72168 C1ZF5V 71549692 IC50 = 180 nM T72168 C15JLF 71549694 IC50 = 120 nM T72168 CUX57Y 71549702 IC50 = 200 nM T72168 CQX42S 71549703 IC50 = 190 nM T72168 CZ3C8X 71549705 IC50 = 500 nM T72168 C0IH6J 71549706 IC50 = 170 nM T72168 CZ8Y7O 71549829 IC50 = 40 nM T72168 CPS61I 71549840 IC50 = 37 nM T72168 CC5AU3 71549841 IC50 = 55 nM T72168 CCV90M 71549842 IC50 = 14 nM T72168 CPFL57 71549843 IC50 = 33 nM T72168 CY8SP0 71549969 IC50 = 210 nM T72168 CXP57U 71549980 IC50 = 180 nM T72168 CA64KN 71550109 IC50 = 400 nM T72168 CUG9C6 71550110 IC50 = 30 nM T72168 CK7NS4 71550116 IC50 = 270 nM T72168 COW8K4 71550118 IC50 = 340 nM T72168 C50TXO 71550241 IC50 = 33 nM T72168 CX6JR5 71550242 IC50 = 34 nM T72168 C93KZM 71550243 IC50 = 42 nM T72168 C6WIA2 71550244 IC50 = 120 nM T72168 CX26UJ 71550250 IC50 = 990 nM T72168 C7R1LJ 71550386 IC50 = 800 nM T72168 CMVD92 71550387 IC50 = 150 nM T72168 CUK7A8 71550511 IC50 = 160 nM T72168 CYB2L0 71550527 IC50 = 230 nM T72168 C6XF9J 71550528 IC50 = 370 nM T72168 CJYQ15 71550529 IC50 = 170 nM T72168 CSHT69 71550657 IC50 = 82 nM T72168 CJX19L 71550659 IC50 = 1530 nM T72168 C6SNW1 71550660 IC50 = 130 nM T72168 CU0Q9P 71550799 IC50 = 470 nM T72168 C8SDX6 71550801 IC50 = 68 nM T72168 CK3HZ0 71550802 IC50 = 240 nM T72168 C9QD8V 71726436 IC50 = 300 nM T72168 CKO01U 71726437 IC50 > 40000 nM T72168 CP9M2C 71726438 IC50 = 750 nM T72168 C6TXD3 71726439 IC50 = 450 nM T72168 CP62QW 71726440 IC50 > 40000 nM T72168 CQYH84 71726556 IC50 > 40000 nM T72168 C8N4UF 71726557 IC50 > 40000 nM T72168 C6TXF5 71726558 IC50 = 500 nM T72168 C4RY0L 71726559 IC50 = 400 nM T72168 CPL35F 71726560 IC50 = 2900 nM T72168 C07YPM 71726687 IC50 > 40000 nM T72168 C6OQT5 71726688 IC50 > 40000 nM T72168 C7F3PL 71726689 IC50 > 40000 nM T72168 C91RTU 71726690 IC50 > 40000 nM T72168 CAR9T3 71726691 IC50 > 40000 nM T72168 C1E3QT 71726810 IC50 > 10000 nM T72168 CV02SB 71726811 IC50 > 40000 nM T72168 C0OXK4 71726812 IC50 > 40000 nM T72168 CL8Z2I 71726813 IC50 = 250 nM T72168 CWS86Q 71726934 IC50 = 3000 nM T72168 C62XFJ 71726935 IC50 > 10000 nM T72168 CIR49D 71726936 IC50 > 40000 nM T72168 CMO7T2 71726937 IC50 = 13000 nM T72168 CE67IF 71726938 IC50 = 16000 nM T72168 CEI4R9 71726939 IC50 > 40000 nM T72168 CKFV04 71727059 IC50 = 2500 nM T72168 CEK6Y8 71727060 IC50 = 1500 nM T72168 CJ0Z6D 71727061 IC50 = 3000 nM T72168 CAG0M9 71727062 IC50 = 300 nM T72168 CN4TI1 71727063 IC50 = 4000 nM T72168 CB45XH 71727183 IC50 = 15000 nM T72168 C76QBF 71727184 IC50 > 40000 nM T72168 CIY4W8 71727185 IC50 > 40000 nM T72168 CB12CL 71727731 IC50 = 6000 nM T72168 C91POE 71727732 IC50 = 1000 nM T72168 C6O2YB 71727733 IC50 = 300 nM T72168 CIUT23 71727734 IC50 = 1000 nM T72168 CE6GH7 71727735 IC50 = 500 nM T72168 CDME45 71727852 IC50 = 3000 nM T72168 C8W7UV 71727853 IC50 = 200 nM T72168 CLTX21 71727854 IC50 = 280 nM T72168 CG0Y6I 71727855 IC50 = 400 nM T72168 C6A1KB 71727856 IC50 = 2600 nM T72168 CRS9A7 71727980 IC50 = 570 nM T72168 CRC7E9 71727981 IC50 = 500 nM T72168 CCK75S 71727982 IC50 > 10000 nM T72168 C3X0QV 71727983 IC50 = 3000 nM T72168 C2KIM1 71727984 IC50 = 600 nM T72168 CKQN54 71728108 IC50 = 2000 nM T72168 C2W9HE 71728109 IC50 = 1000 nM T72168 CVL7Q6 71728110 IC50 = 100 nM T72168 CM78AL 71728111 IC50 = 300 nM T72168 CN80TQ 71728112 IC50 = 100 nM T72168 CF52OE 71728113 IC50 = 4000 nM T72168 C8BGF3 71728224 IC50 = 1200 nM T72168 CJ4M6P 71728225 IC50 = 2000 nM T72168 C10AOX 71728227 IC50 > 30000 nM T72168 C4XSM7 71728228 IC50 = 3000 nM T72168 CW5C6N 71728229 IC50 = 280 nM T72168 CP5KM8 72163477 IC50 = 660 nM T72168 CA6O4K 72163478 IC50 = 750 nM T72168 C27XWS 72163479 IC50 = 1200 nM T72168 C6M9CN 72163480 IC50 = 120 nM T72168 CL8AH4 72163481 IC50 = 550 nM T72168 CB2SD9 72163621 IC50 = 1200 nM T72168 CU6NA8 72163622 IC50 = 170 nM T72168 CTEV75 72163623 IC50 = 33 nM T72168 CER73F 72163624 IC50 = 68 nM T72168 CC8VM7 72163625 IC50 = 1600 nM T72168 CS69AC 72163626 IC50 = 94 nM T72168 CAJ0H5 72163627 IC50 = 43 nM T72168 C1D3EU 72163754 IC50 = 92 nM T72168 C1G3ES 72163755 IC50 = 23 nM T72168 CP8AC2 72188914 EC50 > 5000000 nM T72168 CA6FO5 72188915 EC50 > 5000000 nM T72168 CZ5O6M 72204151 IC50 = 3500 nM T72168 CGT02E 72204156 IC50 = 10900 nM T72168 CW6I9L 72204538 EC50 = 4100 nM T72168 CH5Q8D 72544150 IC50 = 40 nM T72168 C4YUD1 72544151 IC50 = 45 nM T72168 CTM6Y0 72544152 IC50 = 2029 nM T72168 C2K7JR 72544153 IC50 = 1393 nM T72168 C0ZGC8 72544374 IC50 = 1530 nM T72168 CC64LQ 72544375 IC50 = 1974 nM T72168 CNG1C6 72544376 IC50 = 4698 nM T72168 CS1QT2 72544377 IC50 = 121 nM T72168 C0X6YV 72544378 IC50 = 1207 nM T72168 C97CRH 72544379 IC50 = 342 nM T72168 CJ8N2H 72544380 IC50 = 1844 nM T72168 CRB36F 72544601 IC50 = 2086 nM T72168 C3LJ6V 72544602 IC50 = 627 nM T72168 C34FBN 72544603 Ki = 113 nM T72168 CLA3Y9 72710581 Ki = 6.1 nM T72168 CXB45U 72724690 IC50 = 270 nM T72168 CI2K6C 72725442 IC50 = 700 nM T72168 C0W2UD 72725443 IC50 = 400 nM T72168 CQ5D1B 72725444 IC50 = 1100 nM T72168 C2PJV7 72725445 IC50 > 10000 nM T72168 CQ4Z2C 72725446 IC50 = 350 nM T72168 C47IMQ 72725447 IC50 = 2400 nM T72168 CJSK52 72725491 IC50 = 360 nM T72168 CS6J4T 72725492 IC50 = 400 nM T72168 C41FYD 72725493 IC50 = 150 nM T72168 CUG96L 72725494 IC50 = 190 nM T72168 CFHJ16 72725495 IC50 = 400 nM T72168 CW7IY3 72725496 IC50 = 330 nM T72168 CSV1I7 72725497 IC50 = 240 nM T72168 COV09R 72725548 IC50 = 320 nM T72168 CTE01I 72725549 IC50 = 1400 nM T72168 C09ZFS 72725550 IC50 = 480 nM T72168 C2Z7QT 72725551 IC50 = 110 nM T72168 C0K2CP 72725552 IC50 = 5200 nM T72168 C37MEN 72725553 IC50 = 1000 nM T72168 CYSM01 72725554 IC50 = 2300 nM T72168 COU49R 76314656 IC50 = 170 nM T72168 C95NBT 76314657 IC50 > 2000 nM T72168 CL95NP 76317025 IC50 = 609 nM T72168 CZ08OF 76317198 IC50 = 510 nM T72168 CR5B2V 76317199 IC50 = 470 nM T72168 C5YFZ6 76318225 IC50 > 2000 nM T72168 C0RK5D 76321918 IC50 = 1100 nM T72168 C3IC5B 76329113 IC50 > 2000 nM T72168 C1RB6X 76329114 IC50 = 260 nM T72168 CP8M1Z 76332766 IC50 > 2000 nM T72168 CKDI18 76332767 IC50 > 2000 nM T72168 CK21EY 77461202 IC50 = 420 nM T72168 CX20VN 84429708 Ki = 1000 nM T72168 CIU65X 86280440 Ki = 1580 nM T72168 CH46CP 87361539 Ki = 0.08 nM T72168 CT50AL 87539277 IC50 > 1000 nM T72168 CY05IC 87733533 IC50 > 1000 nM T72168 C9EH7I 89500376 Ki > 7010 nM T72168 C0EQS7 89501406 Ki = 415 nM T72168 CG67BU 89508836 IC50 = 130 nM T72168 CBLU18 89509944 IC50 = 380 nM T72168 C8JG7O 89510193 Ki = 1840 nM T72168 CK5D1A 90395281 IC50 = 220 nM T72168 CPC47K 90396922 IC50 = 1600 nM T72168 CQ06RH 90654508 IC50 = 1300 nM T72168 CY5L7N 90655674 IC50 = 660 nM T72168 C9B0QF 90655675 IC50 = 1320 nM T72168 CG6QP2 90655676 IC50 = 670 nM T72168 C8EH0K 90655677 IC50 = 6740 nM T72168 C8GQ4S 90655678 IC50 = 270 nM T72168 C6VZ7X 90656360 IC50 = 9 nM T72168 CNCB43 90656361 IC50 = 10.7 nM T72168 CS42NY 90656362 IC50 = 30.7 nM T72168 C2ZF7W 110763791 Ki = 630.96 nM T72168 CD7RS9 118599615 Ki = 3.981 nM T72168 C70AOV 118599714 Ki = 63.1 nM T72168 C8XLO9 118599727 EC50 = 12.59 nM T72168 CYCM67 118599740 IC50 > 10000 nM T72168 CW7G4T 118599742 Ki = 2.512 nM T72168 C9L5EW 118599756 Ki = 158.49 nM T72168 CVIW94 118599769 EC50 = 1 nM T72168 CFS28Y 118599779 Ki = 50.12 nM T72168 CLS7C1 118707978 EC50 > 5000 nM T72168 C9LV0M 118707979 EC50 > 5000 nM T72168 CC2H4E 118714881 IC50 = 710 nM T72168 C2MQ3P 118714882 IC50 > 10000 nM T72168 CE3I9T 118723172 IC50 > 2000 nM T72168 C13AIC 118723173 IC50 > 2000 nM T72168 C21SWI 118723174 IC50 > 2000 nM T72168 CKR24J 118723175 IC50 > 2000 nM T72168 C28YZF 118723176 IC50 > 2000 nM T72168 C6AGI7 118723177 IC50 > 2000 nM T72168 C4QO8E 118723178 IC50 > 2000 nM T72168 C1RYW9 118796369 Ki = 2 nM T72168 C0X8SA 122178358 IC50 = 1200 nM T72168 C14KFA 122178359 IC50 = 420 nM T72168 C04DIU 122178360 IC50 = 62 nM T72168 CG13LX 122178361 IC50 = 39 nM T72168 C40DRP 122178362 IC50 = 120 nM T72168 C6IV5P 122178363 IC50 = 36 nM T72168 C3MLD0 122178364 IC50 = 64 nM T72168 C0NEZ7 122178365 IC50 = 72 nM T72168 CIT71M 122178366 IC50 = 150 nM T72168 C5ON0U 122178367 IC50 = 1100 nM T72168 C9LIR4 122179356 Ki = 337 nM T72168 CUI57B 122179357 Ki > 3000 nM T72168 CY18QG 122186737 Ki = 2120 nM T72168 C0OR2H 122186738 Ki = 6530 nM T72168 CU0Y8B 122186739 Ki = 3890 nM T72168 CWF0Q4 122186740 Ki = 38.4 nM T72168 CBE6Q8 122186741 Ki = 3880 nM T72168 CX13DR 122186742 Ki = 4250 nM T72168 CJ74HX 122186743 Ki = 3920 nM T72168 C05VWL 122186744 Ki = 44.7 nM T72168 CNX5H4 122186745 Ki = 4470 nM T72168 CQ6BG8 122186747 Ki = 2.1 nM T72168 CH8O2M 122186748 Ki = 27.4 nM T72168 C4LRN1 122186749 Ki = 225 nM T72168 CCK36V 127029882 Ki = 6 nM T72168 CVC84H 127029883 Ki = 6 nM T72168 CFY1P0 127029884 Ki = 6 nM T72168 CU1S6C 127029885 Ki = 7 nM T72168 CA1J0H 127030193 Ki = 1080 nM T72168 CU8Y7N 127030224 Ki = 31 nM T72168 CTEA14 127030225 IC50 = 56 nM T72168 CQ74CG 127030810 Ki = 162 nM T72168 CS5JP0 127031149 Ki = 694 nM T72168 CBW17G 127031150 Ki = 13 nM T72168 C19DUV 127031151 Ki = 14 nM T72168 CLDC46 127031152 Ki = 19 nM T72168 C60SMC 127031153 Ki = 16 nM T72168 C21UAK 127032030 Ki = 144 nM T72168 CBT43F 127032031 Ki = 258 nM T72168 C8TG9C 127032032 Ki = 980 nM T72168 CKZ3X7 127032033 Ki = 55 nM T72168 C8SOU3 127032034 Ki = 230 nM T72168 C87NBI 127032035 Ki = 1452 nM T72168 CKA18M 127032339 Ki > 10 nM T72168 CBR31K 127033260 Ki = 20 nM T72168 CAN7K2 127034410 IC50 = 5217 nM T72168 CSC7I2 127034411 Ki = 1092 nM T72168 C9TG2N 134137487 IC50 > 1000 nM T72168 CTF0J3 135567449 Ki = 1.995 nM T72168 CN24YZ 135567451 EC50 = 0.05012 nM T72168 CPF3B4 135567452 Ki = 0.631 nM T72168 C5MXO2 136000568 Ki > 10000 nM T72168 CM6OX5 136000656 Ki = 2700 nM T72168 CZ2D6U 136059148 Ki = 1600 nM T72168 C6HOU3 136059149 Ki = 1040 nM T72168 CE1G9O 136059150 Ki = 1700 nM T72168 C7LSN6 136088946 Ki = 2800 nM T72168 C3SE8T 136216705 IC50 = 700 nM T72168 CZXM35 136216706 IC50 = 900 nM T72168 CX8H9R 137632028 IC50 = 3900 nM T72168 C0XZC3 137633972 IC50 = 1400 nM T72168 COI80Z 137634236 IC50 > 1000 nM T72168 CP2C7M 137635745 IC50 = 55 nM T72168 CPD87Y 137639726 IC50 > 1000 nM T72168 C3K6DU 137640356 IC50 = 4600 nM T72168 CHTB16 137642739 IC50 = 900 nM T72168 C7KIR1 137643684 IC50 = 6.2 nM T72168 C0J8FI 137646168 IC50 = 4800 nM T72168 CPNB08 137646648 Ki = 195.7 nM T72168 C30ZJF 137648477 IC50 > 1000 nM T72168 C7IG3B 137649694 IC50 = 25 nM T72168 CX63RY 137650280 IC50 = 900 nM T72168 CXWF54 137652695 IC50 = 1100 nM T72168 C69ECN 137653076 IC50 = 18 nM T72168 C8OP2T 137653676 IC50 = 2200 nM T72168 CO92KL 137654415 IC50 > 1000 nM T72168 C8PR9K 137654628 IC50 = 33.4 nM T72168 CX65AR 137656053 IC50 = 1400 nM T72168 CS29XF 137656107 Ki <= 10 nM T72168 C0PL8V 137658165 IC50 = 7 nM T72168 C9GQB2 137658303 IC50 = 1600 nM T72168 C5T7IK 147930449 Ki = 3.981 nM T72168 CCDV87 155511242 IC50 = 114 nM T72168 C28RHM 155514304 Ki = 125.89 nM T72168 CE2YJ9 155514399 Ki = 10 nM T72168 CQF09V 155516050 Ki = 50.12 nM T72168 CQ2GH0 155517818 IC50 = 6309.57 nM T72168 CELU49 155517819 IC50 > 10000 nM T72168 C2E4XV 155518137 Ki = 1000 nM T72168 C4QAB0 155518139 Ki = 1258.93 nM T72168 CCO0Z4 155519877 Ki = 10 nM T72168 C8BD6Y 155522508 Ki = 12.59 nM T72168 CILC13 155524288 IC50 = 5940 nM T72168 C71VIK 155525344 EC50 = 12.59 nM T72168 C1WAQ6 155527406 Ki = 199.53 nM T72168 C5T2QN 155528866 IC50 = 100 nM T72168 CBO7E4 155528935 Ki = 501.19 nM T72168 CQM89D 155529443 Ki < 0.3162 nM T72168 CR0N3F 155529454 Ki = 7.943 nM T72168 CB0XS4 155529625 IC50 > 10000 nM T72168 CLC65H 155532000 Ki = 1995.26 nM T72168 C3HFZ6 155534085 IC50 > 10000 nM T72168 CF52DM 155535034 Ki = 0.5012 nM T72168 CXR2W1 155536089 IC50 = 22 nM T72168 C3FON4 155537084 Ki = 398.11 nM T72168 CUI53F 155537601 Ki = 794.33 nM T72168 C78ISM 155540009 IC50 = 567 nM T72168 CIAW80 155544156 IC50 = 21990 nM T72168 C76OVS 155544396 Ki = 1000 nM T72168 CR6UY8 155545121 IC50 = 20 nM T72168 CE3VY8 155550102 Ki = 6309.57 nM T72168 C6H2ML 155552723 Ki = 7.943 nM T72168 CW8BH4 155554673 Ki = 39.81 nM T72168 C9WV3L 155556878 Ki = 15.85 nM T72168 CR5ZI2 155557239 IC50 = 63.1 nM T72168 CPY83L 155558503 IC50 > 10000 nM T72168 CFAN82 155561077 Ki = 63.1 nM T72168 CQ7HG2 155561626 Ki = 3.162 nM T72168 CXQ23E 155562099 IC50 = 7690 nM T72168 CD4K6Z 155564467 Ki = 0.3162 nM T72168 CS25QB 155564604 IC50 = 32 nM T72168 C7YK6N 155565026 IC50 = 64 nM T72168 C4XJU2 155565054 Ki = 501.19 nM T72168 CPX2J5 155566857 Ki > 6309.57 nM T72168 C79WFJ 155567245 IC50 > 10000 nM T72168 CME1B7 155567676 Ki = 316.23 nM T72168 D00ZGW 46883841 EC50 > 10000 nM T72168 D01ETZ 261000 Ki = 0.54 nM T72168 D01NVD 46830196 EC50 > 19952.62 nM T72168 D04UDT 10407950 IC50 = 126 nM T72168 D07KWO 9823099 IC50 = 6300 nM T72168 D08KQM 24816375 Ki = 149 nM T72168 D09OKK 9951771 IC50 < 20 nM T72168 D0F1SS 44605900 IC50 > 3000000 nM T72168 D0G5OV 11543746 IC50 = 3700 nM T72168 D0M0RS 11560224 Ki > 1000 nM T72168 D0V4RZ 25113722 IC50 > 10000 nM T72168 D0XS0R 44433505 Ki = 124 nM T79724 CN5K3J 135431076 IC50 = 440 nM T79724 C1TGP7 135468747 IC50 = 254000 nM T79724 C64HZJ 135515794 IC50 = 44000 nM T79724 C2WH1V 135526726 IC50 = 139000 nM T79724 CRWV49 135526727 IC50 = 79000 nM T79724 C5R1IQ 135548073 IC50 = 64000 nM T79724 CNLH72 135566603 IC50 > 100000 nM T79724 CAM19I 135566867 IC50 = 51000 nM T79724 CXVR19 135566868 IC50 = 243000 nM T79724 COD4V0 136058510 IC50 = 3160 nM T79724 C2LOX7 136266900 IC50 = 9530 nM T79724 C4OFH6 136610105 IC50 = 82000 nM T79724 CQT2Y1 136610106 IC50 = 88000 nM T49102 D0K8KX 5280343 IC50 = 5730 nM T49102 D0R0MW 5329102 IC50 = 12000 nM T49102 D0E3TC 44259 IC50 = 345 nM T49102 D0Q9CY 9915743 IC50 = 274 nM T49102 D0S3PO 6445562 IC50 = 661 nM T49102 D03BNU 59604787 IC50 > 10000 nM T49102 C8IAR2 5281657 IC50 > 100000 nM T49102 CI68PW 5283685 IC50 > 100000 nM T49102 CXK0S6 5283727 IC50 > 100000 nM T49102 C4G9WR 9547398 IC50 > 100000 nM T49102 C76CUP 9547698 IC50 > 100000 nM T49102 CR8DA1 10024683 IC50 > 100000 nM T49102 CLA93G 10047202 IC50 > 100000 nM T49102 C3LCH5 10047545 IC50 > 100000 nM T49102 C4CP7K 10423452 IC50 = 83900 nM T49102 C83QWV 10714343 IC50 = 14700 nM T49102 C8G5WP 11210533 IC50 = 3780 nM T49102 CBOP58 11293798 Ki > 10000 nM T49102 C26BZX 11362471 Ki > 10000 nM T49102 CWXB93 11397177 Ki > 10000 nM T49102 CL7X4Q 11530963 IC50 > 100000 nM T49102 CTG83F 11539329 Ki > 9200 nM T49102 CACS26 11561968 Ki > 2000 nM T49102 CMIL86 11590363 Ki > 9200 nM T49102 C9T6SC 11640926 Ki > 9200 nM T49102 CU0E8O 11690457 Ki > 2000 nM T49102 CB0AP2 11705863 Ki > 10000 nM T49102 CFPW41 16007116 Ki > 9200 nM T49102 CW2XK6 16050925 IC50 = 25 nM T49102 C5VPH9 16129448 IC50 > 10000 nM T49102 C7YG1N 24759534 IC50 = 16000 nM T49102 CY8L7E 24896769 IC50 > 10000 nM T49102 CLZ23U 24951610 IC50 = 9500 nM T49102 C6BWZ8 25145145 IC50 > 100 nM T49102 C78YWA 25145716 IC50 > 500 nM T49102 C3VRO9 44557921 IC50 > 10000 nM T49102 CY3HW5 46224684 IC50 > 10000 nM T49102 CLS29B 46872626 IC50 > 10000 nM T49102 C2O8RZ 46886323 IC50 = 310 nM T49102 CAH52N 46926529 IC50 = 16900 nM T49102 CF3C9Q 46926532 IC50 = 1300 nM T49102 CKLN53 46926533 IC50 = 1200 nM T49102 CJ0TR2 46926534 IC50 = 710 nM T49102 CZ3XP5 46926535 IC50 = 870 nM T49102 C9VH5T 46931216 IC50 = 4200 nM T49102 CKSN45 49837054 IC50 = 1900 nM T49102 CXR71S 49837055 IC50 = 1900 nM T49102 C9PXN4 49837160 IC50 = 19800 nM T49102 CRT14V 49837161 IC50 = 7800 nM T49102 CEV07X 49837162 IC50 = 48500 nM T49102 C0LIK3 49837163 IC50 > 50000 nM T49102 CZV49T 49837164 IC50 = 18300 nM T49102 CDL7M5 49837165 IC50 = 5700 nM T49102 CGE01R 49837267 IC50 > 50000 nM T49102 CHVJ96 49837268 IC50 = 26200 nM T49102 CJL0X6 49837368 IC50 = 390 nM T49102 CW12AJ 49837369 IC50 = 10800 nM T49102 CB8VJ4 49837370 IC50 = 2700 nM T49102 CNI0A5 49837371 IC50 = 1500 nM T49102 CC8KQ6 49837372 IC50 = 11300 nM T49102 COS6W7 49837473 IC50 = 11200 nM T49102 C0JQD4 49837474 IC50 = 38300 nM T49102 C0R4BG 49837475 IC50 = 1200 nM T49102 CB5D8Q 49837476 IC50 = 1400 nM T49102 CUG43B 49837477 IC50 = 5900 nM T49102 CW8GS0 49837478 IC50 = 5400 nM T49102 C80FJU 49837565 IC50 = 3400 nM T49102 C6KYE4 49837566 IC50 = 7200 nM T49102 CM89FH 49837567 IC50 = 4300 nM T49102 C75GBE 49837568 IC50 = 1900 nM T49102 C42ACM 49837569 IC50 = 1600 nM T49102 CM8LD4 49837570 IC50 = 3400 nM T49102 CN4F3J 50990893 IC50 = 1180 nM T49102 CLO87M 50990894 IC50 = 360 nM T49102 C9MF0X 51355153 IC50 = 5430 nM T49102 COR06H 51355154 IC50 = 6570 nM T49102 C5E7UN 51355155 IC50 = 64400 nM T49102 CPLQ60 51355435 IC50 = 86000 nM T49102 CWJ46U 51355436 IC50 > 50000 nM T49102 CF1D9W 51355713 IC50 = 230 nM T49102 CDT46W 51355977 IC50 = 380 nM T49102 C9ZN0G 51355978 IC50 = 2560 nM T49102 C9TS6F 51355979 IC50 = 4860 nM T49102 CZ82JE 51357926 IC50 = 660 nM T49102 CXA03W 52920796 IC50 > 100 nM T49102 C6OTY5 53251320 IC50 = 13000 nM T49102 CQW5Z9 53262909 IC50 = 770 nM T49102 C0TD7C 53310125 IC50 = 20000 nM T49102 C21FZM 53310126 IC50 = 60 nM T49102 C80WNO 53310127 IC50 = 20 nM T49102 C7DU6V 53310128 IC50 = 130 nM T49102 CBPY13 53310130 IC50 = 4900 nM T49102 CSOD53 53310131 IC50 > 20000 nM T49102 CRV17Y 53310267 IC50 = 620 nM T49102 C4AQN2 53310268 IC50 = 390 nM T49102 CZ78NS 53310269 IC50 > 20000 nM T49102 CAE63S 53310270 IC50 > 20000 nM T49102 CE8OY2 53317913 IC50 > 100 nM T49102 CIN3E9 53318794 IC50 = 200 nM T49102 C0SWH5 53348216 IC50 > 40000 nM T49102 CVG90B 53389651 IC50 > 10000 nM T49102 C9ZFS1 54764923 IC50 > 100000 nM T49102 CIV57W 56947168 IC50 = 2700 nM T49102 CR16SD 56947170 IC50 = 22 nM T49102 C84DVX 57386035 IC50 = 73 nM T49102 CP68IC 57386289 IC50 = 790 nM T49102 C16TMA 57386290 IC50 = 2470 nM T49102 CQCO74 57386291 IC50 = 2680 nM T49102 C57YMK 57386292 IC50 = 2630 nM T49102 C3R7OP 57386802 IC50 = 59 nM T49102 CACW05 57386803 IC50 = 120 nM T49102 C42HDB 57386804 IC50 = 210 nM T49102 CNCO01 57386805 IC50 = 47 nM T49102 CPD52N 57386806 IC50 = 47 nM T49102 CAK54T 57387050 IC50 = 58 nM T49102 CCD90L 57387051 IC50 = 93 nM T49102 CR09GT 57387052 IC50 = 318 nM T49102 CJ1ZP4 57387053 IC50 = 9000 nM T49102 CLW5F4 57387054 IC50 = 10500 nM T49102 CQ60RB 57387300 IC50 = 2260 nM T49102 CG14VM 57387301 IC50 = 1800 nM T49102 C6BPR2 58985201 IC50 > 30000 nM T49102 CXJ63M 59603829 IC50 > 100000 nM T49102 CQEU96 59603842 IC50 = 950 nM T49102 C1MR8Q 60097495 IC50 > 1000 nM T49102 CK6WO0 66552478 IC50 < 10000 nM T49102 CBA0S2 66555775 IC50 = 2000 nM T49102 C37NKO 67129970 IC50 > 10000 nM T49102 CK80LJ 67130050 IC50 > 10000 nM T49102 CV63UL 67240318 IC50 = 1830 nM T49102 C2ZLY3 68310278 IC50 > 100000 nM T49102 C7GRV2 68755406 IC50 > 10000 nM T49102 C5DGR9 69036886 IC50 = 10000 nM T49102 CKT60L 71455860 Ki > 9200 nM T49102 CVIA91 71553085 IC50 = 30000 nM T49102 C1TR3O 71553152 IC50 = 30000 nM T49102 C3UC9H 73891099 IC50 = 1830 nM T49102 CV8QX0 76310169 IC50 = 11800 nM T49102 CA5L4W 76324771 IC50 > 30000 nM T49102 C9GO0P 76328313 IC50 = 6550 nM T49102 CJ2T9E 76332983 IC50 > 10000 nM T49102 C39FTZ 76335685 IC50 > 100000 nM T49102 C1HW4B 89735655 IC50 = 13000 nM T49102 CAU45T 91971978 IC50 > 30000 nM T49102 CU60YC 135431661 IC50 = 1040 nM T49102 CZ7EX0 136183413 IC50 = 3220 nM T49102 CXC69T 137321158 IC50 = 268 nM T49102 CI1E8V 137634241 IC50 > 10000 nM T49102 CXPB85 137634280 IC50 = 808 nM T49102 C7EKT0 137635344 IC50 = 2170 nM T49102 CWG93C 137636215 IC50 = 591 nM T49102 C8GQD5 137636872 IC50 = 1 nM T49102 C8I1KV 137637358 IC50 = 3 nM T49102 C71XKP 137637722 IC50 = 3210 nM T49102 CCT6N8 137637759 IC50 = 197000 nM T49102 CE9RP1 137638267 IC50 = 10000 nM T49102 CX0H1D 137640438 IC50 = 11190 nM T49102 CPZB92 137641994 IC50 = 10030 nM T49102 CBJL60 137643418 IC50 = 87 nM T49102 C3O6XZ 137644537 IC50 = 7 nM T49102 CAFN63 137647467 IC50 = 10030 nM T49102 CCX6Y4 137647984 IC50 = 1600 nM T49102 CJ15KU 137648637 IC50 = 927 nM T49102 C63YRC 137648843 IC50 = 1190 nM T49102 CJW85V 137649497 IC50 = 2400 nM T49102 CYP5X4 137651645 IC50 = 1037 nM T49102 C28QUP 137652864 IC50 > 10000 nM T49102 CU3QA4 137652960 IC50 = 42600 nM T49102 C9MX8B 137653063 IC50 > 10000 nM T49102 C8NR7Y 137654876 IC50 > 200000 nM T49102 C4PGS6 137656550 IC50 = 386 nM T49102 CYB4U5 137658783 IC50 = 1300 nM T49102 COSX73 137659379 IC50 = 478 nM T49102 C41LYM 137659636 IC50 = 838 nM T49102 C4F2EU 137661538 IC50 = 19280 nM T49102 CDNC31 145967951 IC50 > 500 nM T49102 C2MD1Q 155513187 IC50 > 10000 nM T49102 C3LC9I 155536820 IC50 = 1995.26 nM T49102 D00ERW 44444843 Ki > 9242 nM T49102 D00HVA 11624601 Ki > 920 nM T49102 D09LPL 5329103 IC50 = 8000 nM T49102 D0C3KE 16662746 IC50 < 6 nM T49102 D0K0UJ 49837564 IC50 = 230 nM T49102 D0O6OH 71553154 IC50 = 2510 nM T49102 D0Q3NG 11715520 Ki > 920 nM T49102 D0S7IE 11658882 Ki > 9200 nM T49102 D0X1RH 16051023 IC50 = 21 nM T94400 D01XYJ 35370 Ki = 28000 nM T94400 D03KXY 18343 Ki = 560000 nM T94400 D05RHI 6256 Ki = 97000 nM T94400 D05NDN 33039 Ki = 28000 nM T94400 CP25DX 65049 Ki = 238000 nM T94400 C6Q8YR 65311 Ki = 12000 nM T94400 C18KRL 108074 Ki = 230000 nM T94400 C3PLH9 159498 Ki = 122000 nM T94400 C5S6EZ 162501 Ki = 235000 nM T94400 C28WTR 237953 Ki = 75000 nM T94400 C06AIN 451456 Ki = 7000 nM T94400 C5FS1E 477012 Ki = 40000 nM T94400 CL1K7I 477014 Ki = 770000 nM T94400 CI0S8N 477015 Ki = 45000 nM T94400 C9WC1N 499784 Ki = 27000 nM T94400 CDTM30 499785 Ki = 55000 nM T94400 CEA64K 499786 Ki = 19000 nM T94400 C71SME 499787 Ki = 43000 nM T94400 C5Y7SG 502268 Ki = 140000 nM T94400 C1ISO2 502269 Ki = 270000 nM T94400 CLJ46H 502270 Ki = 150000 nM T94400 CN4A5U 508215 Ki = 57000 nM T94400 CZCE20 508216 Ki = 393000 nM T94400 CO9RJ8 510135 Ki = 15000 nM T94400 C82ZIW 510142 Ki = 156000 nM T94400 C72WMJ 510571 Ki = 28000 nM T94400 CZJ7G9 510573 Ki = 90000 nM T94400 C85VPB 510574 Ki = 490000 nM T94400 CX1Y8D 510575 Ki = 1900000 nM T94400 C53QAO 510576 Ki = 140000 nM T94400 CYV0J5 1471774 IC50 = 1900 nM T94400 CFJ5Y3 2743463 IC50 = 3600 nM T94400 CVY6X7 2823137 Ki = 980000 nM T94400 CMV7C0 2823141 Ki = 810000 nM T94400 CVO3D5 3000254 Ki >= 100000 nM T94400 CZF20L 3006428 Ki = 10000 nM T94400 CW0B1Q 3006429 Ki = 10500 nM T94400 CB1UY3 3006430 Ki = 29000 nM T94400 CS6LK5 3006431 Ki = 116000 nM T94400 CMY59Q 3006432 Ki = 315000 nM T94400 C20DTL 5273624 Ki = 390000 nM T94400 CAR3H8 5273625 Ki = 165000 nM T94400 CF85UP 5273627 Ki = 80000 nM T94400 CDM6R5 5273630 Ki = 29000 nM T94400 C2A9TY 5276657 Ki = 89000 nM T94400 CXJ92Z 5276658 Ki = 55000 nM T94400 CS84RK 5276659 Ki = 44000 nM T94400 C7SR0T 5276660 Ki = 45000 nM T94400 CTJH27 5276661 Ki = 90000 nM T94400 C3M1YA 5276662 Ki = 67000 nM T94400 CN5YK8 5276663 Ki = 50000 nM T94400 CQE49Z 5276664 Ki = 44000 nM T94400 CA34BV 5276665 Ki = 38000 nM T94400 C76MVB 5276666 Ki = 195000 nM T94400 C3OQ8G 5276671 Ki = 265000 nM T94400 CI05GN 5276672 Ki = 13000 nM T94400 CQB8D0 5276673 Ki = 10000 nM T94400 CO9LH2 5276674 Ki = 32000 nM T94400 C8FGU9 5713068 IC50 = 634000 nM T94400 C1BF5V 9837976 Ki = 41000 nM T94400 C2E3PN 10084322 Ki = 26500 nM T94400 C7A4CI 10220987 Ki = 6000 nM T94400 CRU39J 10890299 IC50 > 50000 nM T94400 C6K2XY 11162286 Ki = 13500 nM T94400 C53MCF 11483804 Ki = 3500 nM T94400 CJQB38 11500752 Ki = 6500 nM T94400 CYPW14 11523470 Ki = 39000 nM T94400 C5EQ3J 11536969 Ki = 58000 nM T94400 C0R7PJ 11567378 Ki = 19500 nM T94400 C08OBP 11589013 Ki = 38000 nM T94400 C8ZK1F 11594927 Ki = 39000 nM T94400 C4CW2U 11616826 Ki = 96000 nM T94400 CA8PE1 11645614 Ki = 26500 nM T94400 CYBG62 11689746 Ki = 34000 nM T94400 CMU0Q9 11694923 Ki = 51000 nM T94400 CWPA63 11695998 Ki = 23000 nM T94400 CX2U4J 11709208 Ki = 39000 nM T94400 CV82QI 11709226 Ki = 112000 nM T94400 CO04HN 12230213 IC50 = 7700 nM T94400 CM4F6W 12412402 IC50 > 50000 nM T94400 C0PHT1 14606828 Ki = 4200 nM T94400 CRQ1W3 16726539 Ki = 202000 nM T94400 C5PC3K 19093685 IC50 = 133000 nM T94400 CK6Y5F 19093772 IC50 = 590000 nM T94400 C80LTC 19656784 IC50 = 2630 nM T94400 C3DS9Z 23119029 Ki = 70000 nM T94400 CHIC32 23634629 Ki = 16000 nM T94400 CU9F3C 23634630 Ki = 10000 nM T94400 CFD21N 23634631 Ki = 600 nM T94400 CE95YS 23634632 Ki = 15000 nM T94400 C8V1SO 23634745 Ki = 4900 nM T94400 CM6NP9 23634746 Ki = 3800 nM T94400 C1FEL0 23634747 Ki = 1100 nM T94400 CP4NZ2 23634748 Ki = 2300 nM T94400 C9LFB6 23634749 Ki = 35000 nM T94400 CHR0Q2 23635981 Ki = 69000 nM T94400 C5T4BG 23635982 Ki = 21000 nM T94400 CA0B3R 23635983 Ki = 46000 nM T94400 CW96DO 23635984 Ki = 36000 nM T94400 CIS4V6 23635985 Ki = 7200 nM T94400 CAY7H4 23635986 Ki = 12000 nM T94400 CM0L8O 23636103 Ki = 3200 nM T94400 C2UV4C 23636104 Ki = 7800 nM T94400 CNWK28 23636105 Ki = 1000 nM T94400 CP13QF 23636106 Ki = 19200 nM T94400 CCO38E 23636222 Ki = 5400 nM T94400 CJ2ZL1 23636223 Ki = 7200 nM T94400 C0W5RP 23636224 Ki = 2600 nM T94400 CL08SJ 23636225 Ki = 2200 nM T94400 CCX0H8 23636226 Ki = 1900 nM T94400 C89PLD 23636227 Ki = 3800 nM T94400 CKB0A1 23636348 Ki = 260000 nM T94400 CC10EY 23636349 Ki = 37000 nM T94400 C49LUZ 23636479 Ki = 5000 nM T94400 CV3XU0 24764256 Ki = 55000 nM T94400 C5X2YB 44334249 Ki = 5000 nM T94400 C4S9HB 44421254 Ki = 37000 nM T94400 C4YNZ1 44421255 Ki = 180000 nM T94400 C5QB0L 44436021 Ki = 37000 nM T94400 C74ZXQ 44436031 Ki = 15000 nM T94400 C7X0RN 44436053 Ki = 18000 nM T94400 CJ6A8L 44436054 Ki = 5400 nM T94400 C75VRQ 44436073 Ki = 26000 nM T94400 CDV17X 44586051 Ki = 75000 nM T94400 CO0TL1 44586251 Ki = 16000 nM T94400 CI7A8R 44586252 Ki = 35000 nM T94400 CPOH31 44586292 Ki = 26000 nM T94400 C7V9PR 44586335 Ki = 59000 nM T94400 C1ZN0T 44586749 Ki = 52000 nM T94400 C1PCR5 46884564 Ki = 2100 nM T94400 C8DP0M 46885250 Ki = 9900 nM T94400 CQWV32 46885301 Ki = 2700 nM T94400 CUR4G7 46913823 Ki = 18000 nM T94400 C2FX0H 49771519 Ki = 2800 nM T94400 CF1OR6 51034161 Ki = 45000 nM T94400 C5QOM8 51034271 Ki = 2300 nM T94400 CRTC47 53316598 Ki = 1160 nM T94400 CYM4X5 53317249 Ki = 7070 nM T94400 C1REV4 53317250 Ki = 570 nM T94400 CXI90N 53318537 Ki = 930 nM T94400 CPW5E9 53319227 Ki = 270 nM T94400 C7EVS9 53321156 Ki = 5800 nM T94400 CX1J7R 53321424 Ki = 300 nM T94400 CW4Q6N 53323834 Ki = 2460 nM T94400 C6K7ZS 53324520 Ki = 420 nM T94400 C0L1BJ 56656556 Ki = 170 nM T94400 CNH01C 57391914 Ki = 15000 nM T94400 CP5F8G 57393641 Ki = 14500 nM T94400 CZIO94 57395360 Ki = 73000 nM T94400 CT4GF6 57395804 Ki = 201000 nM T94400 C40OJR 57397190 Ki = 35000 nM T94400 CM04OS 57400578 Ki = 9000 nM T94400 C1VH9Q 71508217 Ki = 340000 nM T94400 C64SQB 71508267 Ki = 240000 nM T94400 C12FTK 71508268 Ki = 48000 nM T94400 C1BX3J 71508269 Ki = 70000 nM T94400 C4TZ9O 91801127 IC50 = 420 nM T94400 CZL20I 91801128 IC50 = 2 nM T94400 C2KYI4 91801130 IC50 = 200 nM T94400 C16GEN 101455744 IC50 = 18000 nM T94400 C3FH8V 118725935 IC50 = 1900 nM T94400 C29SWF 118725936 IC50 = 1500 nM T94400 C80FVD 118725937 IC50 = 2730 nM T94400 C5M2ND 118725938 IC50 = 1010 nM T94400 CNT0M2 118725939 IC50 = 1200 nM T94400 CTP48H 118725940 IC50 = 250 nM T94400 C2F9ME 118725941 IC50 = 430 nM T94400 C9H4KS 118725942 IC50 = 8000 nM T94400 CQ3M6O 118725943 IC50 = 14300 nM T94400 C2I1JV 118725944 IC50 = 1200 nM T94400 CX52BM 118725945 IC50 = 6 nM T94400 CJP2F3 118725946 IC50 = 6 nM T94400 C0XB8J 118725947 IC50 = 3 nM T94400 CS5R0M 118725978 IC50 = 5 nM T94400 C6GSK8 118725979 IC50 = 1 nM T94400 CE30HS 118725980 IC50 = 17 nM T94400 C60TWE 118725981 IC50 = 2 nM T94400 CTUA63 118725982 IC50 = 5 nM T94400 C1X8DN 118725983 IC50 = 350 nM T94400 CYE52M 118725984 IC50 = 1000 nM T94400 C5KRC9 118725985 IC50 = 2100 nM T94400 CRCO61 118725986 IC50 = 820 nM T94400 CE85HQ 118725987 IC50 = 240 nM T94400 CI8CG0 118725988 IC50 = 140 nM T94400 C42IWP 118725989 IC50 = 100 nM T94400 CK2E1G 118725990 IC50 = 330 nM T94400 C9TJM4 118725991 IC50 = 22 nM T94400 C7Y3OK 118725992 IC50 = 32 nM T94400 C32HLM 118725993 IC50 > 25000 nM T94400 C2FCR1 118725994 IC50 = 30000 nM T94400 D01GLG 5789 Ki = 27000 nM T94400 D04BBF 447202 Ki = 30000 nM T94400 D0A2IQ 65374 Ki = 10000 nM T94400 D0I9ZJ 447206 Ki = 110000 nM T94400 D0K6QS 65510 Ki = 10000 nM T94400 D0M4MA 6035 Ki = 5000 nM T94400 D0P2IN 27469877 Ki = 16000 nM T94400 D0X1ZP 9427 Ki = 521000 nM T94400 D0Y4MD 66377 Ki = 1140000 nM T94400 D0ZH0I 9700 Ki = 4500 nM T69541 D04DJN 10635 IC50 = 360 nM T69541 D07BSQ 5994 IC50 = 14 nM T69541 D0D1SG 5755 EC50 = 0.002 nM T69541 D0EP0C 5833 IC50 = 1.6 nM T69541 D0G8BV 6450278 Ki = 37 nM T69541 D0I1LH 5839 EC50 = 0.18 nM T69541 D0IT2G 5743 Ki = 0.36 nM T69541 D0Q4SD 443872 IC50 = 63.1 nM T69541 D0Y7IU 5281004 EC50 = 4.8 nM T69541 D0Y7JU 9854489 IC50 = 166 nM T69541 D0Z4EI 55245 IC50 = 590 nM T69541 D00JFE 56941241 IC50 > 1000 nM T69541 D01SYU 10026128 IC50 = 10000 nM T69541 D05RZE 42636651 Ki = 0.33 nM T69541 D07MON 5311505 IC50 = 470 nM T69541 D0SZ1G 121248172 IC50 > 38000 nM T69541 D0X9YP 67041274 IC50 > 10000 nM T69541 D0TH6M 25204767 EC50 > 10000 nM T69541 D0W1XE 91827457 IC50 > 10000 nM T69541 D02KAU 46871935 IC50 = 9 nM T69541 D03KTE 16750192 Ki > 10000 nM T69541 D09UFV 24825740 IC50 > 5000 nM T69541 D0W5RL 9577221 IC50 = 1600 nM T69541 C59UQE 6279 IC50 = 1197 nM T69541 C2O8KM 101788 EC50 = 50 nM T69541 C40YBS 444036 IC50 = 149 nM T69541 C8AMD7 2848661 IC50 = 460 nM T69541 CLBV35 3699263 IC50 = 850 nM T69541 C43BVE 3816305 IC50 = 1070 nM T69541 CDCK27 5185174 IC50 = 1400 nM T69541 C16ZSG 6439929 Ki = 39 nM T69541 C7REX1 9805004 IC50 = 38 nM T69541 CV87EA 9820084 IC50 = 290 nM T69541 C8A3WG 9820510 Ki > 10000 nM T69541 C06RXB 9821393 Ki = 1682 nM T69541 CD9S5P 9825465 Ki = 3838 nM T69541 CE62WD 9839013 IC50 > 1000 nM T69541 CBS8M2 9839134 IC50 = 2369 nM T69541 C92CPK 9841404 Ki > 10000 nM T69541 CK7UC3 9841413 Ki > 10000 nM T69541 C7P6XH 9842832 Ki > 10000 nM T69541 C7RS9U 9846657 Ki > 5000 nM T69541 CERF28 9861044 Ki > 10000 nM T69541 C3K4EU 9862027 Ki > 10000 nM T69541 CEM27C 9885473 IC50 = 3000 nM T69541 C6B9CZ 9888873 IC50 = 160 nM T69541 CZ5R9B 9890023 Ki = 493 nM T69541 CJ7U3R 9904286 IC50 > 10000 nM T69541 C6SWK1 9904610 IC50 = 2492 nM T69541 CTI1J8 9905296 Ki > 10000 nM T69541 CE1TK2 9908041 IC50 > 10000 nM T69541 CMJG42 9921530 IC50 > 10000 nM T69541 C39EXP 9933936 IC50 = 454 nM T69541 C24FUO 9943699 IC50 = 1386 nM T69541 CCSX75 9949772 IC50 = 1500 nM T69541 CKU64T 9952569 IC50 = 333 nM T69541 CW0ED9 9953456 IC50 = 681 nM T69541 C95CAN 9978625 Ki = 0.967 nM T69541 C1QP8T 9993897 IC50 = 2000 nM T69541 C4V6RF 9998996 IC50 > 5000 nM T69541 CC4WY6 10024990 IC50 = 1000 nM T69541 CSM0W3 10026120 IC50 > 2000 nM T69541 CFY67M 10070808 IC50 = 2219 nM T69541 C9T4HR 10071810 IC50 = 1100 nM T69541 CQ3LD1 10091351 IC50 = 1600 nM T69541 C16HAK 10094808 IC50 > 2000 nM T69541 CR0DX5 10126475 IC50 > 1130 nM T69541 CHS18G 10126476 IC50 > 2000 nM T69541 CR0BP6 10126871 IC50 = 380 nM T69541 CV5PQ0 10126940 IC50 = 500 nM T69541 CVF40M 10127159 IC50 = 350 nM T69541 C3CRZ1 10127269 IC50 = 450 nM T69541 CPB60D 10127340 IC50 = 760 nM T69541 CKMW98 10128037 IC50 = 585 nM T69541 C1GI3D 10150743 IC50 = 220 nM T69541 CZKF71 10150825 IC50 = 400 nM T69541 CYR0U5 10150851 IC50 > 2000 nM T69541 CVO1F7 10151165 IC50 = 405 nM T69541 C6EC1P 10151186 IC50 = 405 nM T69541 CQ14RM 10151357 IC50 = 535 nM T69541 CW4Y2K 10151995 IC50 = 1650 nM T69541 C0MX7K 10157532 IC50 = 893 nM T69541 CL0U4N 10172897 IC50 = 400 nM T69541 CG0VH8 10173354 IC50 = 1250 nM T69541 CU6D8W 10173525 IC50 = 170 nM T69541 C8L7HJ 10179031 IC50 = 683 nM T69541 C41YRZ 10194268 IC50 > 740 nM T69541 CX4F7Z 10194607 IC50 > 2000 nM T69541 CV0LE4 10194889 IC50 > 1000 nM T69541 C3O7WH 10215978 IC50 = 1350 nM T69541 C1SG4N 10216152 IC50 > 1420 nM T69541 CD0YT7 10216465 IC50 = 940 nM T69541 C1FGX9 10216535 IC50 = 415 nM T69541 CW7QX2 10216536 IC50 = 720 nM T69541 CG9OH4 10216697 IC50 = 1050 nM T69541 CXN4W1 10216788 IC50 = 1100 nM T69541 CUGN98 10217411 IC50 = 910 nM T69541 CJ9BE0 10222329 IC50 = 651 nM T69541 C84SRT 10223610 IC50 = 2154 nM T69541 CUYO17 10237223 IC50 > 1300 nM T69541 CWYK62 10238100 IC50 = 435 nM T69541 C1R8GY 10238297 IC50 = 900 nM T69541 CNB1V3 10238624 IC50 = 190 nM T69541 CPGF94 10238831 IC50 > 2000 nM T69541 C2AZH1 10238961 IC50 = 175 nM T69541 CSA4R3 10252455 IC50 > 2000 nM T69541 C7EGH2 10252527 IC50 = 120 nM T69541 CR59SC 10271193 IC50 = 22897 nM T69541 CPIS57 10271557 IC50 = 2252 nM T69541 CUQC81 10287415 IC50 > 1000 nM T69541 C5RC7X 10287444 IC50 = 510 nM T69541 CJT2G8 10287863 IC50 = 1400 nM T69541 C1M6WY 10288006 IC50 = 320 nM T69541 CO6UP3 10288155 IC50 = 875 nM T69541 C6C2IK 10288565 IC50 = 195 nM T69541 CNEO49 10289020 IC50 = 104 nM T69541 CLJU03 10298892 Ki = 3914 nM T69541 C9UYG8 10309447 IC50 > 1050 nM T69541 C8FM2D 10309755 IC50 = 1800 nM T69541 C1OV7M 10309756 IC50 = 715 nM T69541 C9TI4A 10310063 IC50 = 1035 nM T69541 CP9AE0 10310476 IC50 > 512 nM T69541 CV52EN 10310809 IC50 = 140 nM T69541 CR1L5N 10311251 IC50 = 104 nM T69541 CX7WS4 10316069 IC50 = 354 nM T69541 CQP1Y7 10340204 IC50 = 1525 nM T69541 CEJ78I 10365592 IC50 > 2000 nM T69541 CDBZ06 10372181 IC50 = 120 nM T69541 C14AIB 10384345 IC50 = 970 nM T69541 CZ5CJ3 10423330 IC50 > 10000 nM T69541 C5I3BG 10428464 Ki = 12 nM T69541 C1KE6C 10446402 IC50 = 2050 nM T69541 C0NT9D 10454007 IC50 > 5000 nM T69541 C85RBN 10474264 IC50 > 2000 nM T69541 CUL8O4 10475384 IC50 > 5000 nM T69541 CPX65M 10477088 IC50 = 130 nM T69541 C5AP6C 10503520 IC50 > 10000 nM T69541 CBEC38 10596252 IC50 = 1000 nM T69541 CC8T7J 10598305 IC50 = 1062 nM T69541 CO3V0S 10622594 IC50 = 977 nM T69541 C02ZMG 10643956 IC50 = 748 nM T69541 CYNG45 10668755 IC50 > 10000 nM T69541 CYRQ10 10691647 Ki = 1100 nM T69541 CVD2Y9 10717098 IC50 > 10000 nM T69541 CAT1X8 10741366 IC50 = 1068 nM T69541 CB3JD0 10763832 IC50 = 1358 nM T69541 C07BOR 10787258 IC50 = 2035 nM T69541 C1CRQ5 10811045 IC50 > 10000 nM T69541 CN1H5Z 10832792 IC50 = 1592 nM T69541 CHU9A4 10873317 IC50 = 334 nM T69541 CHU10G 10960295 IC50 = 1850 nM T69541 C6LYG7 11090322 IC50 > 1000 nM T69541 CXS6J7 11155441 Ki = 10 nM T69541 CQUV78 11176984 IC50 = 23 nM T69541 CL97OU 11212803 IC50 = 540 nM T69541 C4U0DF 11213029 Ki = 980 nM T69541 CRN4V2 11232136 IC50 > 3000 nM T69541 C8XPZ4 11269445 IC50 > 2000 nM T69541 C4HNB8 11269886 IC50 = 1050 nM T69541 CC0XI4 11279959 IC50 = 440 nM T69541 C4SC0W 11281576 IC50 > 5000 nM T69541 C8YL6K 11282486 IC50 = 1700 nM T69541 CUX0S2 11282904 Ki = 21 nM T69541 CIY9H5 11291999 IC50 = 1800 nM T69541 C0IQ9K 11304445 IC50 = 160 nM T69541 C0XUF2 11305564 IC50 > 5000 nM T69541 CXC9G3 11327341 IC50 > 2000 nM T69541 CT9Y4O 11339440 IC50 = 2300 nM T69541 C8FQ9B 11375180 IC50 = 21000 nM T69541 CP2DL0 11377050 IC50 = 1000 nM T69541 C76VYN 11382721 IC50 > 2000 nM T69541 CV4RO2 11384310 IC50 = 48 nM T69541 CXW40M 11384346 IC50 > 2000 nM T69541 CU7IE0 11410199 IC50 = 690 nM T69541 CO20QH 11416730 IC50 = 155 nM T69541 C5WO0U 11429662 IC50 > 5000 nM T69541 CD2Q3F 11474917 IC50 = 83 nM T69541 CC75NQ 11477616 Ki = 430 nM T69541 CQ62KS 11485693 IC50 > 3000 nM T69541 C9Q1NY 11494167 Ki = 32 nM T69541 CFLQ08 11495227 IC50 = 320 nM T69541 C03NYX 11495549 IC50 = 90 nM T69541 CR40IH 11516847 IC50 = 1800 nM T69541 CP4F8X 11517412 IC50 = 280 nM T69541 C2PB6Z 11530605 Ki = 930 nM T69541 C1R6DC 11531942 IC50 = 140 nM T69541 CZ1HA3 11538472 IC50 = 615 nM T69541 CFC1Z4 11538799 IC50 = 1100 nM T69541 CBK60G 11559947 IC50 > 2000 nM T69541 C1D9YS 11560003 IC50 > 2000 nM T69541 CB37YF 11566981 Ki = 145 nM T69541 C8WJ2F 11567609 IC50 = 780 nM T69541 C0SCT6 11588584 IC50 = 810 nM T69541 C3MW1D 11589982 IC50 = 220 nM T69541 C03QYZ 11590471 IC50 = 110 nM T69541 CAO2P1 11596392 IC50 > 2000 nM T69541 CSB97O 11617028 Ki = 21 nM T69541 CRL3A7 11632925 IC50 = 120 nM T69541 CQB0E3 11633482 IC50 = 65 nM T69541 C9DNG1 11640164 IC50 = 580 nM T69541 C1RJ3I 11646689 IC50 = 1000 nM T69541 CX3L5S 11647533 IC50 = 80 nM T69541 C4S5RG 11655053 IC50 = 175 nM T69541 CDOZ32 11661172 IC50 = 590 nM T69541 C0LEZ3 11667800 Ki = 890 nM T69541 C5XEN0 11668719 IC50 = 220 nM T69541 CZPK72 11682989 IC50 = 80 nM T69541 CCK83U 11690269 IC50 = 160 nM T69541 CY07JH 11696378 IC50 > 2000 nM T69541 CBU02W 11696959 IC50 = 640 nM T69541 C2S9IT 11697271 IC50 = 1900 nM T69541 CGR32I 11697882 IC50 = 340 nM T69541 C75IBX 11704529 IC50 = 90 nM T69541 CGX54N 11704756 IC50 = 210 nM T69541 CO2N1W 11710364 IC50 = 1550 nM T69541 CZ52YQ 11710766 IC50 < 500 nM T69541 C8OPA1 11710962 IC50 = 855 nM T69541 CW3N8H 11711766 IC50 = 280 nM T69541 COEU05 11719039 IC50 = 100 nM T69541 CZ0B7H 11731863 IC50 = 1900 nM T69541 CQO76Z 11741168 IC50 > 2000 nM T69541 C87YNC 11741891 IC50 = 150 nM T69541 CH92VI 11743259 IC50 = 310 nM T69541 C5HLU8 11750204 IC50 = 380 nM T69541 CY1F4I 11752649 Ki = 670 nM T69541 CQU0E7 11774868 IC50 = 435 nM T69541 C4U8KY 12085089 IC50 = 162 nM T69541 C14LTD 15463551 IC50 > 1000 nM T69541 C3QOV0 16099227 IC50 = 430 nM T69541 CW6LO1 16099229 IC50 > 2000 nM T69541 C2R4PK 16099231 IC50 = 450 nM T69541 C9KM7X 16099232 IC50 = 1900 nM T69541 C05CYN 16099234 IC50 = 1600 nM T69541 CJQ8A1 16099236 IC50 = 450 nM T69541 CA72YW 16099237 IC50 > 2000 nM T69541 CS07DB 16099238 IC50 = 98 nM T69541 C42ESN 16099240 IC50 = 580 nM T69541 CMZ91J 16099242 IC50 > 2000 nM T69541 CF69RC 16099243 IC50 > 2000 nM T69541 C60GEM 16099245 IC50 = 1500 nM T69541 CE48CS 16099246 IC50 = 620 nM T69541 CTF2M7 16099247 IC50 = 130 nM T69541 CX9BK2 16099248 IC50 = 775 nM T69541 CN6PA9 16099249 IC50 = 350 nM T69541 C9Z6AK 16099250 IC50 = 120 nM T69541 C5Z8HR 16099251 IC50 = 91 nM T69541 CWK76M 16099252 IC50 = 880 nM T69541 C3BU9M 16216822 IC50 = 290 nM T69541 C1Q5SV 16220168 IC50 = 510 nM T69541 CH6CN0 16658901 Ki > 10000 nM T69541 CU9LS2 16661702 EC50 = 5000 nM T69541 C1UY8J 16666386 IC50 > 1000 nM T69541 CWK35C 16730429 IC50 = 8700 nM T69541 CSKX58 17758233 Ki = 410 nM T69541 C7CPW9 17758234 Ki = 48 nM T69541 CI5KT6 17758236 Ki = 42 nM T69541 C3FP7L 17921933 IC50 = 3162 nM T69541 CX03YG 18188955 IC50 = 1220 nM T69541 CR19ST 18512166 IC50 = 310 nM T69541 CEN14G 18512334 IC50 = 4000 nM T69541 CS9CI5 18551230 IC50 = 30 nM T69541 CBI64N 18551237 IC50 = 130 nM T69541 C5ZYJ0 20231824 Ki = 952 nM T69541 CEH7V5 20786216 IC50 > 1000 nM T69541 C97WCO 21941658 IC50 = 1.259 nM T69541 CCI89R 21948853 IC50 > 1000 nM T69541 CB2SF4 21948904 IC50 > 1000 nM T69541 C2ZP7V 22218142 IC50 = 1500 nM T69541 C1QTK4 22398492 IC50 = 240 nM T69541 C6CSB4 22398502 IC50 > 2000 nM T69541 CR8N1E 22398506 IC50 = 1420 nM T69541 CM83TU 22398533 IC50 = 265 nM T69541 C34LHW 22398559 IC50 = 910 nM T69541 CJBW90 22398592 IC50 > 2000 nM T69541 CEJ65O 22398627 IC50 = 415 nM T69541 CZI4C6 24739672 Ki = 1000 nM T69541 CS23KY 24739834 Ki = 1390 nM T69541 C1M9QG 24739836 Ki = 1770 nM T69541 CG5SJ0 24739997 Ki = 1490 nM T69541 C7Z1HW 24740156 Ki = 1440 nM T69541 CTE1N2 24748569 EC50 > 10000 nM T69541 C4WYE7 24749678 Ki = 1.56 nM T69541 CY2JS4 24749684 Ki = 1.51 nM T69541 C2QHO3 24749808 Ki = 0.319 nM T69541 C5S6JN 24780149 IC50 > 1000 nM T69541 CW5TJ7 24781731 IC50 > 1000 nM T69541 C1JTW2 24851053 Ki = 0.342 nM T69541 CC53XL 24860583 Ki > 3000 nM T69541 C58RHY 24883011 IC50 = 80 nM T69541 CW35CK 24883012 IC50 = 41 nM T69541 C3SC0V 24883054 IC50 = 76 nM T69541 C4SA6C 24883055 IC50 = 15 nM T69541 C5LZK2 24895096 IC50 = 1350 nM T69541 COGP96 24936313 IC50 > 5000 nM T69541 CVY09S 24936449 IC50 > 5000 nM T69541 C06PDG 24952192 EC50 > 5000 nM T69541 CG1CF9 24952193 EC50 > 5000 nM T69541 CZC7L8 24953162 IC50 > 10000 nM T69541 C4W7BN 24954947 IC50 > 10000 nM T69541 C6XC2R 24954951 IC50 > 20000 nM T69541 CYES17 24957737 Ki > 3000 nM T69541 C83YKB 24961057 Ki > 1000 nM T69541 CIGM27 24983460 IC50 = 280 nM T69541 CHY0D7 25013322 IC50 > 10000 nM T69541 C0TPS5 25013653 IC50 > 10000 nM T69541 CWU91M 25013811 IC50 > 10000 nM T69541 CSH29L 25013812 IC50 > 10000 nM T69541 C7QCX0 25052023 IC50 = 2.4 nM T69541 CAW8M0 25070694 IC50 = 2800 nM T69541 C21XDY 25145083 Ki > 10000 nM T69541 CS6JQ1 25167502 Ki = 155 nM T69541 C0XPW9 25168896 IC50 = 340 nM T69541 CUL27D 25168900 IC50 = 260 nM T69541 CEV2D7 25205475 IC50 = 260 nM T69541 C9S0ZW 25205477 IC50 = 330 nM T69541 C49KHR 25206116 IC50 = 510 nM T69541 C9FM2U 42642501 Ki <= 10 nM T69541 CXZ35T 44193145 Ki = 656 nM T69541 C2MOF7 44193146 Ki = 378 nM T69541 CWR6X1 44193147 Ki = 2250 nM T69541 C3JOW4 44193245 Ki = 1470 nM T69541 CHGI03 44251606 IC50 = 475 nM T69541 C0OA6M 44264483 IC50 > 10000 nM T69541 COCE32 44264569 IC50 > 10000 nM T69541 CI0TN2 44264577 IC50 > 10000 nM T69541 CXOR54 44264579 IC50 > 10000 nM T69541 C01HSQ 44264588 IC50 > 10000 nM T69541 CDB54J 44305270 IC50 > 1000 nM T69541 C0XLN6 44305556 IC50 > 1000 nM T69541 C1UK4M 44305720 IC50 = 1889 nM T69541 CH4PU5 44305819 IC50 = 2484 nM T69541 C6N1AR 44305929 IC50 2871 nM T69541 C73CXK 44354006 IC50 = 363 nM T69541 C0N3TD 44354884 IC50 = 2700 nM T69541 CPQ2A6 44354885 IC50 = 1000 nM T69541 CM0G1V 44354886 IC50 = 2000 nM T69541 CL6G3Q 44355066 IC50 = 2100 nM T69541 CSAU31 44377064 IC50 > 10000 nM T69541 C7H9NC 44377081 IC50 > 10000 nM T69541 C60DYH 44377090 IC50 = 2000 nM T69541 CVH2R3 44377098 IC50 = 2900 nM T69541 CYLI63 44377110 IC50 > 10000 nM T69541 CQX39I 44377356 IC50 = 570 nM T69541 C9FJW4 44377382 IC50 = 1900 nM T69541 C13SYV 44396250 Ki = 300 nM T69541 CB1P0S 44396251 Ki = 80 nM T69541 CHY1C3 44396271 Ki = 590 nM T69541 C29MBI 44396272 Ki = 310 nM T69541 C4TQ6N 44396282 Ki = 440 nM T69541 CH2Y3L 44396283 Ki = 190 nM T69541 CWZB52 44396284 Ki = 850 nM T69541 CD80LM 44396296 Ki > 1000 nM T69541 C6SI5L 44396297 Ki > 1000 nM T69541 CR4H1E 44396316 Ki = 510 nM T69541 C45LRH 44396317 Ki = 140 nM T69541 C5JG6H 44396330 Ki > 1000 nM T69541 CA8V4G 44396331 Ki > 1000 nM T69541 C57CPQ 44396332 Ki = 310 nM T69541 CXHF58 44403036 IC50 = 215 nM T69541 C6JNI4 44403038 IC50 = 60 nM T69541 C45SOW 44403039 IC50 = 315 nM T69541 CXZ4S3 44426781 Ki = 3490 nM T69541 C8HO4K 44426782 Ki = 585 nM T69541 C0FEN3 44426790 Ki = 298 nM T69541 C19MJP 44426793 Ki = 527 nM T69541 C1ZDA4 44426795 Ki = 1270 nM T69541 CIOW01 44431179 IC50 = 520 nM T69541 C3SJ5V 44433504 Ki = 7.5 nM T69541 C2SCP7 44435606 IC50 = 1600 nM T69541 CH5E3L 44435611 IC50 > 1300 nM T69541 CDO62N 44435656 IC50 = 650 nM T69541 C9TP4C 44435662 IC50 = 345 nM T69541 C19TMW 44435663 IC50 = 730 nM T69541 C90WUC 44435667 IC50 = 430 nM T69541 CHFB89 44435668 IC50 = 300 nM T69541 C8IWK2 44435669 IC50 = 250 nM T69541 CYG7X4 44473146 IC50 > 10000 nM T69541 CR5SI0 44476535 EC50 > 10000 nM T69541 CM29JD 44516036 IC50 > 10000 nM T69541 CR19IH 44543858 IC50 > 2000 nM T69541 C05HEP 44543860 IC50 > 2000 nM T69541 C45ZHO 44543969 IC50 > 2000 nM T69541 C25OXZ 44544094 IC50 > 2000 nM T69541 C7JIF6 44544321 IC50 > 2000 nM T69541 CF6V4G 44563171 EC50 > 10000 nM T69541 C8BGL6 44585565 IC50 > 3000 nM T69541 CIJP09 44605898 IC50 > 10000000 nM T69541 C9PLK4 45263610 IC50 > 2000 nM T69541 C78JKD 45265930 IC50 = 1100 nM T69541 C08UBE 45272032 IC50 > 10000 nM T69541 C57EZH 45275745 IC50 = 110 nM T69541 CU7D0O 45278780 IC50 = 3.7 nM T69541 CY8A1D 45278857 IC50 = 3.1 nM T69541 CGX87F 45279098 IC50 = 6.5 nM T69541 CL9P2A 45380783 IC50 = 3.8 nM T69541 CKC0B7 46237842 IC50 = 59 nM T69541 C4KN0J 46237981 IC50 = 31 nM T69541 C7KW8T 46883839 EC50 > 10000 nM T69541 CZSG25 46883893 EC50 > 10000 nM T69541 C72MUY 46889765 IC50 > 5000 nM T69541 C6DVO1 46889848 IC50 > 10000 nM T69541 CZ90FC 46894119 Ki = 9 nM T69541 C04KWS 46913888 IC50 = 54 nM T69541 C1U7QL 46913889 IC50 = 52 nM T69541 C3Q7RI 46913890 IC50 = 6 nM T69541 CY7D0I 46913891 IC50 = 80 nM T69541 CQ93ML 46913892 IC50 = 135 nM T69541 C1ZRD2 46914168 IC50 = 1620 nM T69541 CWV42M 46914169 IC50 = 3740 nM T69541 CK6SJ3 46914453 IC50 = 275 nM T69541 C4HQ5Y 46914584 IC50 = 223 nM T69541 C9F4PR 46914585 IC50 = 4340 nM T69541 CZE49A 46914586 IC50 = 553 nM T69541 CGS9U8 46914587 IC50 = 41 nM T69541 C34EDY 46914588 IC50 = 21 nM T69541 CLCI21 46914734 IC50 = 13 nM T69541 C2NM6E 46914737 IC50 = 25 nM T69541 CKP01L 46914738 IC50 = 58 nM T69541 CP91XE 46914741 IC50 = 89 nM T69541 C3Q5PE 46914742 IC50 = 4 nM T69541 C6OG0A 46914743 IC50 = 7 nM T69541 C1TMA8 46914744 IC50 = 150 nM T69541 CE7KZ8 46914881 IC50 = 83 nM T69541 CI0Y4F 46914882 IC50 > 10000 nM T69541 C8HWO7 46914883 IC50 = 784 nM T69541 C6FN4G 46914884 IC50 = 246 nM T69541 CXY74T 46914885 IC50 = 9730 nM T69541 CF1D5Q 46914886 IC50 = 488 nM T69541 CVGF35 46914887 IC50 > 500 nM T69541 C4ZPR6 46915029 IC50 = 180 nM T69541 CXR29C 46915030 IC50 > 10000 nM T69541 C9NC0K 46915031 IC50 = 1440 nM T69541 CY3O2C 46915043 IC50 = 41 nM T69541 CHG94E 46915044 IC50 = 32 nM T69541 CK85FJ 46915045 IC50 = 101 nM T69541 CQ6J3N 46915201 IC50 = 2080 nM T69541 CC84WO 46915202 IC50 = 8360 nM T69541 CTM2J5 46915203 IC50 = 31 nM T69541 C75IFZ 46915353 IC50 = 16 nM T69541 CJW51A 46915354 IC50 = 26 nM T69541 CX70GY 46915355 IC50 = 15.2 nM T69541 CPTL45 46915356 IC50 = 2 nM T69541 C39SUV 46915640 IC50 = 243 nM T69541 CX6WK5 46915641 IC50 = 535 nM T69541 CW8J2E 46915642 IC50 = 56 nM T69541 C05YTF 46915643 IC50 = 284 nM T69541 CMW7E4 46915644 IC50 = 56 nM T69541 CA43UG 46915645 IC50 > 127 nM T69541 CJ3DN2 46915781 IC50 > 1000 nM T69541 C4L1JF 46915782 IC50 = 383 nM T69541 CB4X3D 46915783 IC50 > 10000 nM T69541 CK7DI0 46915784 IC50 > 10000 nM T69541 CU7L4T 46915785 IC50 = 10000 nM T69541 CE9OU3 46915786 IC50 = 410 nM T69541 CI3E2M 46915787 IC50 = 763 nM T69541 C1BV5K 46916070 IC50 = 3650 nM T69541 C06JHQ 46916071 IC50 = 441 nM T69541 CQ37UY 46916072 IC50 = 1590 nM T69541 C38HIP 46916073 IC50 = 1290 nM T69541 CPK95L 46916074 IC50 = 151 nM T69541 C7NC4B 46917090 IC50 = 2.8 nM T69541 C2LCJ7 46937290 IC50 = 210 nM T69541 CKQ8J3 46937431 IC50 > 2000 nM T69541 CL7P3N 46938234 IC50 = 1.8 nM T69541 COS28G 46938235 IC50 = 18 nM T69541 CFJT93 46938236 IC50 = 7.6 nM T69541 CHL70M 46938239 IC50 = 4.1 nM T69541 C8P7JH 46938914 IC50 > 2000 nM T69541 CY95VK 46938915 IC50 > 2000 nM T69541 CVX25Q 46938916 IC50 = 220 nM T69541 C2V5AT 46939019 IC50 = 480 nM T69541 C5R6GI 46939020 IC50 = 390 nM T69541 CF1BX0 46939115 IC50 > 2000 nM T69541 C4P0EU 46939116 IC50 = 160 nM T69541 CD6B7X 46939395 IC50 = 58 nM T69541 C1KXF2 46939396 IC50 > 2000 nM T69541 CVN4W1 47958757 IC50 = 168 nM T69541 CX0NO8 49782554 EC50 < 15848.93 nM T69541 CC7T8Q 49782555 EC50 < 15848.93 nM T69541 CD07EV 49782777 EC50 < 15848.93 nM T69541 C43UKW 49782778 IC50 < 14421.15 nM T69541 C2JTF0 49782779 EC50 < 15848.93 nM T69541 CS7KX9 49782780 IC50 < 12560.3 nM T69541 C36RYU 49782781 IC50 = 5140.44 nM T69541 C8OA0C 49782985 EC50 < 15848.93 nM T69541 C5Y6QU 49782986 EC50 < 15848.93 nM T69541 CB8V7R 49782987 EC50 < 15848.93 nM T69541 CU3S6H 49836028 EC50 > 5000 nM T69541 C96SLW 49851364 EC50 > 5000 nM T69541 CDN4K6 49851369 EC50 > 5000 nM T69541 C4YXN1 49851467 EC50 > 5000 nM T69541 CUD91T 49862248 EC50 > 10000 nM T69541 C5NX4D 49864061 IC50 = 2530 nM T69541 CPH9D8 49864098 IC50 = 69 nM T69541 CMS1N3 49864127 IC50 = 15 nM T69541 CTE0N7 49864128 IC50 = 720 nM T69541 COP7W2 49864129 IC50 = 127 nM T69541 CCKJ45 49864153 IC50 = 849 nM T69541 C19FRV 49864154 IC50 = 65 nM T69541 CWGD27 49864174 IC50 = 146 nM T69541 C9YCN1 49864175 IC50 = 39 nM T69541 CTKV39 49864176 IC50 = 26 nM T69541 CZ8J1V 50942115 Ki = 800 nM T69541 C23OEF 50942312 EC50 > 10000 nM T69541 CX1KO8 51346768 Ki = 849 nM T69541 C7N9TD 51346823 Ki = 1518 nM T69541 C0WDX3 51347001 Ki = 1115 nM T69541 CF8DK7 51347002 Ki = 3170 nM T69541 CTH45Q 52918523 IC50 > 10000 nM T69541 CL8D1Z 52921432 IC50 = 130 nM T69541 CEC4I7 52941608 IC50 = 230 nM T69541 CDV90J 52942528 IC50 > 1000 nM T69541 C8Y9SU 52944898 IC50 > 1000 nM T69541 CK5UT4 53317489 Ki = 126 nM T69541 CM0LU1 53318659 Ki = 1200 nM T69541 CUD48O 53320087 Ki = 0.64 nM T69541 CD0N1K 53323476 IC50 = 356 nM T69541 CYH3V0 53325642 Ki = 86.8 nM T69541 C82DYI 53326614 Ki > 4170 nM T69541 CJCP75 53359074 EC50 > 5000 nM T69541 C9H5YE 53361128 EC50 > 5000 nM T69541 CUR24K 53875787 IC50 = 2800 nM T69541 C1JR5W 54576068 IC50 = 24 nM T69541 CS62XZ 54590901 IC50 = 53.9 nM T69541 C30XLO 54592009 Ki = 6.3 nM T69541 CCS8R6 54592010 IC50 = 39 nM T69541 CML2E7 54592011 IC50 = 86 nM T69541 CRVB01 54592087 IC50 = 266 nM T69541 C7W1BA 54592088 IC50 = 109 nM T69541 C9N3IS 54592089 IC50 = 56 nM T69541 C2GML6 54592090 IC50 = 33 nM T69541 C05FVP 54592092 IC50 = 19 nM T69541 C9W5DZ 56593984 EC50 > 5000 nM T69541 CF3G2M 56925477 IC50 = 36 nM T69541 CZ7O8G 56925478 IC50 = 69 nM T69541 CV5C0T 56925479 IC50 > 10000 nM T69541 C9ITY0 56925480 IC50 > 10000 nM T69541 C3M4TE 56925570 IC50 = 920 nM T69541 CZ4I2J 56925571 IC50 = 6800 nM T69541 CW87RG 56925573 IC50 = 2000 nM T69541 C4Z5LF 56925574 IC50 = 4100 nM T69541 CKF8Z3 56925575 IC50 = 1300 nM T69541 CY20OR 56925668 IC50 > 10000 nM T69541 C30DAL 56925669 IC50 = 600 nM T69541 CQHA65 56925670 IC50 = 310 nM T69541 CJP31U 56925671 IC50 = 270 nM T69541 CV86DS 56925673 IC50 = 2700 nM T69541 CI3S6F 56925790 IC50 = 5300 nM T69541 CTY1Q9 56925791 IC50 = 1100 nM T69541 CH40YG 56925792 IC50 = 960 nM T69541 C2PLD4 56925793 IC50 = 260 nM T69541 CU02HT 56925794 IC50 = 570 nM T69541 CM19WI 56925904 IC50 > 10000 nM T69541 CA7BX4 56925905 IC50 = 440 nM T69541 CTR7X3 56925906 IC50 = 1100 nM T69541 C39VBK 56925907 IC50 = 430 nM T69541 CV7EN5 56925908 IC50 = 320 nM T69541 CU69SK 56925909 IC50 = 590 nM T69541 CAMI87 56925910 IC50 = 700 nM T69541 CTG9I7 56926011 IC50 = 70 nM T69541 CPD82H 56968080 IC50 = 7.1 nM T69541 CM0SG2 57390990 IC50 = 1100 nM T69541 CU8AN3 57392780 IC50 = 790 nM T69541 CX12JM 57392781 IC50 = 45 nM T69541 C9OMW1 57392782 IC50 = 405 nM T69541 C30JOV 57394501 IC50 = 190 nM T69541 CINU04 57396254 IC50 = 225 nM T69541 C1O6JU 57396255 IC50 = 230 nM T69541 CVOB64 57399718 IC50 = 610 nM T69541 CF83VM 57401459 EC50 > 5000 nM T69541 C7W3YD 57401479 IC50 = 430 nM T69541 CR6L7E 57403222 IC50 = 1450 nM T69541 CPU6W7 57473898 IC50 = 80 nM T69541 CEJ25K 57473899 IC50 = 270 nM T69541 CUJ08D 57474008 IC50 = 70 nM T69541 CDB0F1 57503322 IC50 = 39 nM T69541 CIDS61 57503325 IC50 = 19 nM T69541 C2U1GQ 57524309 IC50 = 22 nM T69541 C0BDS9 57585514 IC50 < 2 nM T69541 CM17UZ 57585515 IC50 = 47 nM T69541 CYGU85 57585534 IC50 = 1.3 nM T69541 C3WG0L 57666312 Ki = 1100 nM T69541 C43GDR 57666397 Ki = 290 nM T69541 CTM6K5 57690900 IC50 > 5000 nM T69541 CB2I7A 57748722 Ki <= 10 nM T69541 CT9Y6X 57748723 Ki <= 10 nM T69541 C6J0HD 57748748 Ki <= 10 nM T69541 C2MFH6 57748755 Ki <= 10 nM T69541 CMR56T 57748765 Ki <= 10 nM T69541 C05UIP 57748768 Ki <= 10 nM T69541 CH2PV6 57748780 Ki = 0.79 nM T69541 CL13HZ 57748781 Ki = 0.4 nM T69541 C7UH3N 57748789 Ki <= 10 nM T69541 C2YT7S 57748790 Ki = 0.23 nM T69541 C1KZT3 57906156 IC50 = 500 nM T69541 C3IN9F 57983276 IC50 = 170 nM T69541 CJ6Y1B 58026134 IC50 > 2000 nM T69541 C19XQV 58026164 IC50 > 2000 nM T69541 CR7H3O 58026170 IC50 > 2000 nM T69541 C7XL3D 58026176 IC50 > 2000 nM T69541 CT1EM3 58064710 IC50 = 3.7 nM T69541 C8S3EQ 58064714 IC50 = 2.7 nM T69541 CPI62D 58064720 IC50 = 2.2 nM T69541 CL42XF 58064726 IC50 = 4.3 nM T69541 CPL9A6 58064729 IC50 = 55.9 nM T69541 CRFS78 58064730 IC50 = 3.3 nM T69541 CN1J3V 58064734 IC50 = 17.8 nM T69541 CA0SH5 58064735 IC50 = 4.4 nM T69541 CI7BP4 58064741 IC50 = 21.4 nM T69541 C2FZA7 58064756 IC50 = 9.4 nM T69541 C3AMO0 58064757 IC50 = 4450 nM T69541 C47AUR 58392644 EC50 = 2.5 nM T69541 C9CQS0 58392665 EC50 = 3.2 nM T69541 CXF39M 58392685 EC50 > 3000 nM T69541 C7FXH3 58392721 EC50 > 3000 nM T69541 CJDN90 58392790 EC50 = 1.6 nM T69541 CO59DQ 58392803 EC50 > 3000 nM T69541 C5K9PJ 58483018 IC50 = 1.2 nM T69541 C4C2FT 58599563 IC50 = 1300 nM T69541 CWAD17 58731166 Ki <= 500 nM T69541 CNE02T 58731180 Ki <= 500 nM T69541 CVS58C 58731199 Ki <= 500 nM T69541 C3VU0Q 58731202 Ki <= 500 nM T69541 C03HFM 58731234 Ki <= 500 nM T69541 CADQ18 58731243 Ki <= 500 nM T69541 CI7XQ5 58731245 Ki <= 500 nM T69541 C67UET 58731323 Ki <= 500 nM T69541 C0JL7A 58973277 IC50 > 1000 nM T69541 CY38HG 59233337 Ki > 1000 nM T69541 CUX4E7 59233347 Ki > 3333 nM T69541 CO63VJ 59233364 Ki > 1000 nM T69541 C2A9JO 59251119 IC50 > 5000 nM T69541 CD8A6P 59281281 IC50 = 49 nM T69541 CBZ0M5 59281312 IC50 = 170 nM T69541 CCT59B 59281329 IC50 = 510 nM T69541 CQI5C4 59281343 IC50 = 38 nM T69541 CH5E1F 59281346 IC50 > 10000 nM T69541 CPE83R 59281354 IC50 = 180 nM T69541 CI9EP1 59281363 IC50 = 8.4 nM T69541 CQ2BO1 59281403 IC50 = 51 nM T69541 CP78RD 59281411 IC50 = 95 nM T69541 CCNU12 59281412 IC50 = 10 nM T69541 C7HVB1 59281416 IC50 = 490 nM T69541 CE5A0V 59281447 IC50 = 75 nM T69541 CZT9S6 59281449 IC50 = 430 nM T69541 CIKQ89 59281508 IC50 = 990 nM T69541 CE1A7J 59281531 IC50 = 680 nM T69541 CK9JZ4 59281538 IC50 = 36 nM T69541 C4TG5U 59281540 IC50 = 22 nM T69541 CPC80S 59281541 IC50 = 64 nM T69541 CXS5C4 59281543 IC50 = 250 nM T69541 C7KPR9 59281566 IC50 = 150 nM T69541 CUJP64 59281599 IC50 = 600 nM T69541 CYZI85 59556974 IC50 > 10000 nM T69541 C5C3AO 59770003 Ki = 2.48 nM T69541 CH36PL 59807625 IC50 < 500 nM T69541 C54ATL 59807726 IC50 < 500 nM T69541 C8S7OB 59808080 IC50 < 500 nM T69541 CYU57B 59808129 IC50 < 500 nM T69541 C2TNO8 60026286 IC50 > 2000 nM T69541 CZE5J8 60026377 IC50 > 2000 nM T69541 C0LDS2 60026592 IC50 = 1150 nM T69541 C31PTC 60026641 IC50 > 2000 nM T69541 C67NSE 60026675 IC50 > 2000 nM T69541 C6GP5R 60026731 IC50 = 720 nM T69541 C5M8HV 60026772 IC50 = 1200 nM T69541 CI36XS 60026787 IC50 > 2000 nM T69541 C3JD8M 60026802 IC50 > 2000 nM T69541 CE9MI4 60026817 IC50 = 1900 nM T69541 C04EKW 60026878 IC50 > 2000 nM T69541 CPRW14 66991384 IC50 = 160 nM T69541 CYP31Z 66995780 IC50 = 3050 nM T69541 CK36QI 66996020 IC50 > 10000 nM T69541 CJ09TZ 66996063 IC50 = 2225 nM T69541 C3EU7N 66996137 IC50 = 276 nM T69541 C1CXY9 66996546 IC50 = 401 nM T69541 C9Y2DN 66996560 IC50 = 727 nM T69541 C9LOZ1 66996568 IC50 = 1181 nM T69541 CH39DP 67053383 IC50 > 2000 nM T69541 C3LF8O 67053425 IC50 > 2000 nM T69541 CMYP75 67415874 IC50 = 100 nM T69541 CQU8E3 68031408 IC50 = 11 nM T69541 C1FK3D 69081573 IC50 = 31 nM T69541 CB6HX8 69082589 IC50 = 480 nM T69541 C43PON 69675755 IC50 = 9.4 nM T69541 COR52G 69675880 IC50 = 13 nM T69541 C9Q7VH 70561849 IC50 = 39 nM T69541 CARO49 70685018 Ki = 150 nM T69541 C5QPC0 70697572 Ki = 170 nM T69541 C94FCP 71452686 IC50 = 3000 nM T69541 CF08ME 71457470 Ki = 0.4 nM T69541 CEO5G4 71461616 IC50 = 1900 nM T69541 C78IOK 71467161 IC50 = 310 nM T69541 C1MHC0 71467246 IC50 = 47 nM T69541 C4B0IC 71467248 IC50 = 26 nM T69541 CYW34A 71519686 IC50 = 120 nM T69541 CGK4S8 71543393 Ki = 1450 nM T69541 C83YJF 71544946 IC50 = 39 nM T69541 CK2O1Z 71545110 IC50 = 54 nM T69541 C0LD8K 71548690 IC50 = 270 nM T69541 C19CGP 71548691 IC50 = 1700 nM T69541 C4BE6G 71548692 IC50 = 1110 nM T69541 CCK7Q3 71548693 IC50 = 240 nM T69541 CK9S0J 71548694 IC50 = 1440 nM T69541 CT9Y5D 71549558 Ki = 2 nM T69541 C8ZX0F 71549573 IC50 = 180 nM T69541 COQ5C4 71549690 IC50 = 230 nM T69541 CE7NZ0 71549691 IC50 = 190 nM T69541 C1ZF5V 71549692 IC50 = 180 nM T69541 C15JLF 71549694 IC50 = 120 nM T69541 CUX57Y 71549702 IC50 = 200 nM T69541 CQX42S 71549703 IC50 = 190 nM T69541 CZ3C8X 71549705 IC50 = 500 nM T69541 C0IH6J 71549706 IC50 = 170 nM T69541 CZ8Y7O 71549829 IC50 = 40 nM T69541 CPS61I 71549840 IC50 = 37 nM T69541 CC5AU3 71549841 IC50 = 55 nM T69541 CCV90M 71549842 IC50 = 14 nM T69541 CPFL57 71549843 IC50 = 33 nM T69541 CY8SP0 71549969 IC50 = 210 nM T69541 CXP57U 71549980 IC50 = 180 nM T69541 CA64KN 71550109 IC50 = 400 nM T69541 CUG9C6 71550110 IC50 = 30 nM T69541 CK7NS4 71550116 IC50 = 270 nM T69541 COW8K4 71550118 IC50 = 340 nM T69541 C50TXO 71550241 IC50 = 33 nM T69541 CX6JR5 71550242 IC50 = 34 nM T69541 C93KZM 71550243 IC50 = 42 nM T69541 C6WIA2 71550244 IC50 = 120 nM T69541 CX26UJ 71550250 IC50 = 990 nM T69541 C7R1LJ 71550386 IC50 = 800 nM T69541 CMVD92 71550387 IC50 = 150 nM T69541 CUK7A8 71550511 IC50 = 160 nM T69541 CYB2L0 71550527 IC50 = 230 nM T69541 C6XF9J 71550528 IC50 = 370 nM T69541 CJYQ15 71550529 IC50 = 170 nM T69541 CSHT69 71550657 IC50 = 82 nM T69541 CJX19L 71550659 IC50 = 1530 nM T69541 C6SNW1 71550660 IC50 = 130 nM T69541 CU0Q9P 71550799 IC50 = 470 nM T69541 C8SDX6 71550801 IC50 = 68 nM T69541 CK3HZ0 71550802 IC50 = 240 nM T69541 C9QD8V 71726436 IC50 = 300 nM T69541 CKO01U 71726437 IC50 > 40000 nM T69541 CP9M2C 71726438 IC50 = 750 nM T69541 C6TXD3 71726439 IC50 = 450 nM T69541 CP62QW 71726440 IC50 > 40000 nM T69541 CQYH84 71726556 IC50 > 40000 nM T69541 C8N4UF 71726557 IC50 > 40000 nM T69541 C6TXF5 71726558 IC50 = 500 nM T69541 C4RY0L 71726559 IC50 = 400 nM T69541 CPL35F 71726560 IC50 = 2900 nM T69541 C07YPM 71726687 IC50 > 40000 nM T69541 C6OQT5 71726688 IC50 > 40000 nM T69541 C7F3PL 71726689 IC50 > 40000 nM T69541 C91RTU 71726690 IC50 > 40000 nM T69541 CAR9T3 71726691 IC50 > 40000 nM T69541 C1E3QT 71726810 IC50 > 10000 nM T69541 CV02SB 71726811 IC50 > 40000 nM T69541 C0OXK4 71726812 IC50 > 40000 nM T69541 CL8Z2I 71726813 IC50 = 250 nM T69541 CWS86Q 71726934 IC50 = 3000 nM T69541 C62XFJ 71726935 IC50 > 10000 nM T69541 CIR49D 71726936 IC50 > 40000 nM T69541 CMO7T2 71726937 IC50 = 13000 nM T69541 CE67IF 71726938 IC50 = 16000 nM T69541 CEI4R9 71726939 IC50 > 40000 nM T69541 CKFV04 71727059 IC50 = 2500 nM T69541 CEK6Y8 71727060 IC50 = 1500 nM T69541 CJ0Z6D 71727061 IC50 = 3000 nM T69541 CAG0M9 71727062 IC50 = 300 nM T69541 CN4TI1 71727063 IC50 = 4000 nM T69541 CB45XH 71727183 IC50 = 15000 nM T69541 C76QBF 71727184 IC50 > 40000 nM T69541 CIY4W8 71727185 IC50 > 40000 nM T69541 CB12CL 71727731 IC50 = 6000 nM T69541 C91POE 71727732 IC50 = 1000 nM T69541 C6O2YB 71727733 IC50 = 300 nM T69541 CIUT23 71727734 IC50 = 1000 nM T69541 CE6GH7 71727735 IC50 = 500 nM T69541 CDME45 71727852 IC50 = 3000 nM T69541 C8W7UV 71727853 IC50 = 200 nM T69541 CLTX21 71727854 IC50 = 280 nM T69541 CG0Y6I 71727855 IC50 = 400 nM T69541 C6A1KB 71727856 IC50 = 2600 nM T69541 CRS9A7 71727980 IC50 = 570 nM T69541 CRC7E9 71727981 IC50 = 500 nM T69541 CCK75S 71727982 IC50 > 10000 nM T69541 C3X0QV 71727983 IC50 = 3000 nM T69541 C2KIM1 71727984 IC50 = 600 nM T69541 CKQN54 71728108 IC50 = 2000 nM T69541 C2W9HE 71728109 IC50 = 1000 nM T69541 CVL7Q6 71728110 IC50 = 100 nM T69541 CM78AL 71728111 IC50 = 300 nM T69541 CN80TQ 71728112 IC50 = 100 nM T69541 CF52OE 71728113 IC50 = 4000 nM T69541 C8BGF3 71728224 IC50 = 1200 nM T69541 CJ4M6P 71728225 IC50 = 2000 nM T69541 C10AOX 71728227 IC50 > 30000 nM T69541 C4XSM7 71728228 IC50 = 3000 nM T69541 CW5C6N 71728229 IC50 = 280 nM T69541 CP5KM8 72163477 IC50 = 660 nM T69541 CA6O4K 72163478 IC50 = 750 nM T69541 C27XWS 72163479 IC50 = 1200 nM T69541 C6M9CN 72163480 IC50 = 120 nM T69541 CL8AH4 72163481 IC50 = 550 nM T69541 CB2SD9 72163621 IC50 = 1200 nM T69541 CU6NA8 72163622 IC50 = 170 nM T69541 CTEV75 72163623 IC50 = 33 nM T69541 CER73F 72163624 IC50 = 68 nM T69541 CC8VM7 72163625 IC50 = 1600 nM T69541 CS69AC 72163626 IC50 = 94 nM T69541 CAJ0H5 72163627 IC50 = 43 nM T69541 C1D3EU 72163754 IC50 = 92 nM T69541 C1G3ES 72163755 IC50 = 23 nM T69541 CP8AC2 72188914 EC50 > 5000000 nM T69541 CA6FO5 72188915 EC50 > 5000000 nM T69541 CZ5O6M 72204151 IC50 = 3500 nM T69541 CGT02E 72204156 IC50 = 10900 nM T69541 CW6I9L 72204538 EC50 = 4100 nM T69541 CH5Q8D 72544150 IC50 = 40 nM T69541 C4YUD1 72544151 IC50 = 45 nM T69541 CTM6Y0 72544152 IC50 = 2029 nM T69541 C2K7JR 72544153 IC50 = 1393 nM T69541 C0ZGC8 72544374 IC50 = 1530 nM T69541 CC64LQ 72544375 IC50 = 1974 nM T69541 CNG1C6 72544376 IC50 = 4698 nM T69541 CS1QT2 72544377 IC50 = 121 nM T69541 C0X6YV 72544378 IC50 = 1207 nM T69541 C97CRH 72544379 IC50 = 342 nM T69541 CJ8N2H 72544380 IC50 = 1844 nM T69541 CRB36F 72544601 IC50 = 2086 nM T69541 C3LJ6V 72544602 IC50 = 627 nM T69541 C34FBN 72544603 Ki = 113 nM T69541 CLA3Y9 72710581 Ki = 6.1 nM T69541 CXB45U 72724690 IC50 = 270 nM T69541 CI2K6C 72725442 IC50 = 700 nM T69541 C0W2UD 72725443 IC50 = 400 nM T69541 CQ5D1B 72725444 IC50 = 1100 nM T69541 C2PJV7 72725445 IC50 > 10000 nM T69541 CQ4Z2C 72725446 IC50 = 350 nM T69541 C47IMQ 72725447 IC50 = 2400 nM T69541 CJSK52 72725491 IC50 = 360 nM T69541 CS6J4T 72725492 IC50 = 400 nM T69541 C41FYD 72725493 IC50 = 150 nM T69541 CUG96L 72725494 IC50 = 190 nM T69541 CFHJ16 72725495 IC50 = 400 nM T69541 CW7IY3 72725496 IC50 = 330 nM T69541 CSV1I7 72725497 IC50 = 240 nM T69541 COV09R 72725548 IC50 = 320 nM T69541 CTE01I 72725549 IC50 = 1400 nM T69541 C09ZFS 72725550 IC50 = 480 nM T69541 C2Z7QT 72725551 IC50 = 110 nM T69541 C0K2CP 72725552 IC50 = 5200 nM T69541 C37MEN 72725553 IC50 = 1000 nM T69541 CYSM01 72725554 IC50 = 2300 nM T69541 COU49R 76314656 IC50 = 170 nM T69541 C95NBT 76314657 IC50 > 2000 nM T69541 CL95NP 76317025 IC50 = 609 nM T69541 CZ08OF 76317198 IC50 = 510 nM T69541 CR5B2V 76317199 IC50 = 470 nM T69541 C5YFZ6 76318225 IC50 > 2000 nM T69541 C0RK5D 76321918 IC50 = 1100 nM T69541 C3IC5B 76329113 IC50 > 2000 nM T69541 C1RB6X 76329114 IC50 = 260 nM T69541 CP8M1Z 76332766 IC50 > 2000 nM T69541 CKDI18 76332767 IC50 > 2000 nM T69541 CK21EY 77461202 IC50 = 420 nM T69541 CX20VN 84429708 Ki = 1000 nM T69541 CIU65X 86280440 Ki = 1580 nM T69541 CH46CP 87361539 Ki = 0.08 nM T69541 CT50AL 87539277 IC50 > 1000 nM T69541 CY05IC 87733533 IC50 > 1000 nM T69541 C9EH7I 89500376 Ki > 7010 nM T69541 C0EQS7 89501406 Ki = 415 nM T69541 CG67BU 89508836 IC50 = 130 nM T69541 CBLU18 89509944 IC50 = 380 nM T69541 C8JG7O 89510193 Ki = 1840 nM T69541 CK5D1A 90395281 IC50 = 220 nM T69541 CPC47K 90396922 IC50 = 1600 nM T69541 CQ06RH 90654508 IC50 = 1300 nM T69541 CY5L7N 90655674 IC50 = 660 nM T69541 C9B0QF 90655675 IC50 = 1320 nM T69541 CG6QP2 90655676 IC50 = 670 nM T69541 C8EH0K 90655677 IC50 = 6740 nM T69541 C8GQ4S 90655678 IC50 = 270 nM T69541 C6VZ7X 90656360 IC50 = 9 nM T69541 CNCB43 90656361 IC50 = 10.7 nM T69541 CS42NY 90656362 IC50 = 30.7 nM T69541 C2ZF7W 110763791 Ki = 630.96 nM T69541 CD7RS9 118599615 Ki = 3.981 nM T69541 C70AOV 118599714 Ki = 63.1 nM T69541 C8XLO9 118599727 EC50 = 12.59 nM T69541 CYCM67 118599740 IC50 > 10000 nM T69541 CW7G4T 118599742 Ki = 2.512 nM T69541 C9L5EW 118599756 Ki = 158.49 nM T69541 CVIW94 118599769 EC50 = 1 nM T69541 CFS28Y 118599779 Ki = 50.12 nM T69541 CLS7C1 118707978 EC50 > 5000 nM T69541 C9LV0M 118707979 EC50 > 5000 nM T69541 CC2H4E 118714881 IC50 = 710 nM T69541 C2MQ3P 118714882 IC50 > 10000 nM T69541 CE3I9T 118723172 IC50 > 2000 nM T69541 C13AIC 118723173 IC50 > 2000 nM T69541 C21SWI 118723174 IC50 > 2000 nM T69541 CKR24J 118723175 IC50 > 2000 nM T69541 C28YZF 118723176 IC50 > 2000 nM T69541 C6AGI7 118723177 IC50 > 2000 nM T69541 C4QO8E 118723178 IC50 > 2000 nM T69541 C1RYW9 118796369 Ki = 2 nM T69541 C0X8SA 122178358 IC50 = 1200 nM T69541 C14KFA 122178359 IC50 = 420 nM T69541 C04DIU 122178360 IC50 = 62 nM T69541 CG13LX 122178361 IC50 = 39 nM T69541 C40DRP 122178362 IC50 = 120 nM T69541 C6IV5P 122178363 IC50 = 36 nM T69541 C3MLD0 122178364 IC50 = 64 nM T69541 C0NEZ7 122178365 IC50 = 72 nM T69541 CIT71M 122178366 IC50 = 150 nM T69541 C5ON0U 122178367 IC50 = 1100 nM T69541 C9LIR4 122179356 Ki = 337 nM T69541 CUI57B 122179357 Ki > 3000 nM T69541 CY18QG 122186737 Ki = 2120 nM T69541 C0OR2H 122186738 Ki = 6530 nM T69541 CU0Y8B 122186739 Ki = 3890 nM T69541 CWF0Q4 122186740 Ki = 38.4 nM T69541 CBE6Q8 122186741 Ki = 3880 nM T69541 CX13DR 122186742 Ki = 4250 nM T69541 CJ74HX 122186743 Ki = 3920 nM T69541 C05VWL 122186744 Ki = 44.7 nM T69541 CNX5H4 122186745 Ki = 4470 nM T69541 CQ6BG8 122186747 Ki = 2.1 nM T69541 CH8O2M 122186748 Ki = 27.4 nM T69541 C4LRN1 122186749 Ki = 225 nM T69541 CCK36V 127029882 Ki = 6 nM T69541 CVC84H 127029883 Ki = 6 nM T69541 CFY1P0 127029884 Ki = 6 nM T69541 CU1S6C 127029885 Ki = 7 nM T69541 CA1J0H 127030193 Ki = 1080 nM T69541 CU8Y7N 127030224 Ki = 31 nM T69541 CTEA14 127030225 IC50 = 56 nM T69541 CQ74CG 127030810 Ki = 162 nM T69541 CS5JP0 127031149 Ki = 694 nM T69541 CBW17G 127031150 Ki = 13 nM T69541 C19DUV 127031151 Ki = 14 nM T69541 CLDC46 127031152 Ki = 19 nM T69541 C60SMC 127031153 Ki = 16 nM T69541 C21UAK 127032030 Ki = 144 nM T69541 CBT43F 127032031 Ki = 258 nM T69541 C8TG9C 127032032 Ki = 980 nM T69541 CKZ3X7 127032033 Ki = 55 nM T69541 C8SOU3 127032034 Ki = 230 nM T69541 C87NBI 127032035 Ki = 1452 nM T69541 CKA18M 127032339 Ki > 10 nM T69541 CBR31K 127033260 Ki = 20 nM T69541 CAN7K2 127034410 IC50 = 5217 nM T69541 CSC7I2 127034411 Ki = 1092 nM T69541 C9TG2N 134137487 IC50 > 1000 nM T69541 CTF0J3 135567449 Ki = 1.995 nM T69541 CN24YZ 135567451 EC50 = 0.05012 nM T69541 CPF3B4 135567452 Ki = 0.631 nM T69541 C5MXO2 136000568 Ki > 10000 nM T69541 CM6OX5 136000656 Ki = 2700 nM T69541 CZ2D6U 136059148 Ki = 1600 nM T69541 C6HOU3 136059149 Ki = 1040 nM T69541 CE1G9O 136059150 Ki = 1700 nM T69541 C7LSN6 136088946 Ki = 2800 nM T69541 C3SE8T 136216705 IC50 = 700 nM T69541 CZXM35 136216706 IC50 = 900 nM T69541 CX8H9R 137632028 IC50 = 3900 nM T69541 C0XZC3 137633972 IC50 = 1400 nM T69541 COI80Z 137634236 IC50 > 1000 nM T69541 CP2C7M 137635745 IC50 = 55 nM T69541 CPD87Y 137639726 IC50 > 1000 nM T69541 C3K6DU 137640356 IC50 = 4600 nM T69541 CHTB16 137642739 IC50 = 900 nM T69541 C7KIR1 137643684 IC50 = 6.2 nM T69541 C0J8FI 137646168 IC50 = 4800 nM T69541 CPNB08 137646648 Ki = 195.7 nM T69541 C30ZJF 137648477 IC50 > 1000 nM T69541 C7IG3B 137649694 IC50 = 25 nM T69541 CX63RY 137650280 IC50 = 900 nM T69541 CXWF54 137652695 IC50 = 1100 nM T69541 C69ECN 137653076 IC50 = 18 nM T69541 C8OP2T 137653676 IC50 = 2200 nM T69541 CO92KL 137654415 IC50 > 1000 nM T69541 C8PR9K 137654628 IC50 = 33.4 nM T69541 CX65AR 137656053 IC50 = 1400 nM T69541 CS29XF 137656107 Ki <= 10 nM T69541 C0PL8V 137658165 IC50 = 7 nM T69541 C9GQB2 137658303 IC50 = 1600 nM T69541 C5T7IK 147930449 Ki = 3.981 nM T69541 CCDV87 155511242 IC50 = 114 nM T69541 C28RHM 155514304 Ki = 125.89 nM T69541 CE2YJ9 155514399 Ki = 10 nM T69541 CQF09V 155516050 Ki = 50.12 nM T69541 CQ2GH0 155517818 IC50 = 6309.57 nM T69541 CELU49 155517819 IC50 > 10000 nM T69541 C2E4XV 155518137 Ki = 1000 nM T69541 C4QAB0 155518139 Ki = 1258.93 nM T69541 CCO0Z4 155519877 Ki = 10 nM T69541 C8BD6Y 155522508 Ki = 12.59 nM T69541 CILC13 155524288 IC50 = 5940 nM T69541 C71VIK 155525344 EC50 = 12.59 nM T69541 C1WAQ6 155527406 Ki = 199.53 nM T69541 C5T2QN 155528866 IC50 = 100 nM T69541 CBO7E4 155528935 Ki = 501.19 nM T69541 CQM89D 155529443 Ki < 0.3162 nM T69541 CR0N3F 155529454 Ki = 7.943 nM T69541 CB0XS4 155529625 IC50 > 10000 nM T69541 CLC65H 155532000 Ki = 1995.26 nM T69541 C3HFZ6 155534085 IC50 > 10000 nM T69541 CF52DM 155535034 Ki = 0.5012 nM T69541 CXR2W1 155536089 IC50 = 22 nM T69541 C3FON4 155537084 Ki = 398.11 nM T69541 CUI53F 155537601 Ki = 794.33 nM T69541 C78ISM 155540009 IC50 = 567 nM T69541 CIAW80 155544156 IC50 = 21990 nM T69541 C76OVS 155544396 Ki = 1000 nM T69541 CR6UY8 155545121 IC50 = 20 nM T69541 CE3VY8 155550102 Ki = 6309.57 nM T69541 C6H2ML 155552723 Ki = 7.943 nM T69541 CW8BH4 155554673 Ki = 39.81 nM T69541 C9WV3L 155556878 Ki = 15.85 nM T69541 CR5ZI2 155557239 IC50 = 63.1 nM T69541 CPY83L 155558503 IC50 > 10000 nM T69541 CFAN82 155561077 Ki = 63.1 nM T69541 CQ7HG2 155561626 Ki = 3.162 nM T69541 CXQ23E 155562099 IC50 = 7690 nM T69541 CD4K6Z 155564467 Ki = 0.3162 nM T69541 CS25QB 155564604 IC50 = 32 nM T69541 C7YK6N 155565026 IC50 = 64 nM T69541 C4XJU2 155565054 Ki = 501.19 nM T69541 CPX2J5 155566857 Ki > 6309.57 nM T69541 C79WFJ 155567245 IC50 > 10000 nM T69541 CME1B7 155567676 Ki = 316.23 nM T69541 D00ZGW 46883841 EC50 > 10000 nM T69541 D01ETZ 261000 Ki = 0.54 nM T69541 D01NVD 46830196 EC50 > 19952.62 nM T69541 D04UDT 10407950 IC50 = 126 nM T69541 D07KWO 9823099 IC50 = 6300 nM T69541 D08KQM 24816375 Ki = 149 nM T69541 D09OKK 9951771 IC50 < 20 nM T69541 D0F1SS 44605900 IC50 > 3000000 nM T69541 D0G5OV 11543746 IC50 = 3700 nM T69541 D0M0RS 11560224 Ki > 1000 nM T69541 D0V4RZ 25113722 IC50 > 10000 nM T69541 D0XS0R 44433505 Ki = 124 nM T94033 D05PHH 3447 IC50 = 687 nM T94033 D07UWV 92722 IC50 = 3.88 nM T94033 D07XHO 4413 IC50 = 1900 nM T94033 D08YIN 1727 Ki > 2000000 nM T94033 D0AZ8C 5213 IC50 = 20900 nM T94033 D0FT4R 107706 IC50 > 2000 nM T94033 D0I0EG 44093 Ki = 48 nM T94033 D0I0RJ 16231 IC50 > 20000 nM T94033 D0I5HF 10182969 Ki = 3100 nM T94033 D0J0BU 10275777 IC50 = 18 nM T94033 D0K8KX 5280343 IC50 = 30000 nM T94033 D0KG3R 9875401 Ki > 1000 nM T94033 D0M7JT 216210 IC50 = 1.2 nM T94033 D0SH3I 387447 Ki = 13000 nM T94033 D0V3YT 10324367 IC50 < 1000 nM T94033 D0X9CH 3010818 IC50 < 1000 nM T94033 D0Y7LD 222284 Ki = 267.2 nM T94033 D00LOB 9866964 Ki = 1.3 nM T94033 D01MUU 183797 Ki = 1.2 nM T94033 D05HAD 9955534 Ki = 5.2 nM T94033 D05TKW 16098914 IC50 = 1100 nM T94033 D05TPI 72276 IC50 = 150000 nM T94033 D08PBB 177992 IC50 = 78760 nM T94033 D0I7MX 9871765 Ki = 0.015 nM T94033 D0ID3W 9911502 Ki = 367 nM T94033 D0K4FP 44548240 IC50 = 150 nM T94033 D0KI5R 135565674 IC50 = 2.63 nM T94033 D0PK7J 56599309 Ki = 9490 nM T94033 D0X2NN 9826322 Ki = 2.7 nM T94033 D0Y6SQ 2536 IC50 = 780 nM T94033 D02INZ 2387 IC50 = 31000 nM T94033 D02MHE 9806376 IC50 = 1.2 nM T94033 D02QTV 122267 IC50 = 0.03 nM T94033 D03QJN 9895762 Ki = 6000 nM T94033 D08ELM 9832212 IC50 = 370 nM T94033 D0D5RH 11641515 IC50 = 1200 nM T94033 D0E2MJ 5496659 Ki > 4000 nM T94033 D0G7YZ 9869699 Ki = 8.17 nM T94033 D0GR2H 11740077 IC50 = 1600 nM T94033 D0H4UJ 66005 Ki = 4.2 nM T94033 D0J9UI 9807238 IC50 = 7.7 nM T94033 D0N7WR 108040 Ki = 2500 nM T94033 D0Q3WN 6918278 Ki = 0.27 nM T94033 D0RP8F 5311176 IC50 = 0.003 ug.mL-1 T94033 D0S2JG 9913629 Ki = 0.38 nM T94033 D0Y5EX 122296 Ki = 0.04 nM T94033 CR8YG3 1308 Ki = 1200 nM T94033 C71WRJ 1503 Ki = 41000 nM T94033 CY5B9C 1504 Ki = 15000 nM T94033 C2KE5Q 1508 Ki = 13000 nM T94033 C2SHL9 1623 Ki = 2.1 nM T94033 CKO7V4 1701 IC50 = 62000 nM T94033 C7BU1L 2138 Ki = 3981.07 nM T94033 C4S1PB 4300 Ki = 245000 nM T94033 CL1T7V 4301 Ki = 22000 nM T94033 C65JEN 4406 IC50 = 690 nM T94033 C8D4SG 5107 Ki > 3000 nM T94033 CRAO91 5324 Ki = 95 nM T94033 C7RE8Y 5738 Ki = 374 nM T94033 CF7IL1 10860 Ki = 1700 nM T94033 CUSM50 11974 Ki = 946 nM T94033 C2OG9Z 47978 IC50 = 5000 nM T94033 C5P3TH 65130 Ki = 224 nM T94033 C9TN2A 75626 Ki = 95000 nM T94033 C2G6KL 87925 Ki = 195 nM T94033 COHM79 117475 Ki = 3162277.66 nM T94033 CMG15V 122129 Ki > 2000 nM T94033 CK9AZ0 122670 IC50 = 22000 nM T94033 CLX4V7 130395 IC50 = 107500 nM T94033 CD14RN 197789 Ki = 39810.72 nM T94033 CZP0Y1 204101 Ki = 540 nM T94033 C2HTG4 229074 Ki = 1995262.31 nM T94033 C2SW0R 270006 IC50 = 330000 nM T94033 C1WRQ6 309231 IC50 >= 30000 nM T94033 CU4G3Y 309369 Ki = 79432.82 nM T94033 CHB2N8 313890 Ki = 320 nM T94033 C4JKM8 313891 Ki = 180 nM T94033 CJ9LT4 347113 IC50 = 20000 nM T94033 CM32OH 402499 IC50 = 7000 nM T94033 C4Q9XJ 402501 IC50 > 50000 nM T94033 CZ1QL5 411406 Ki = 796 nM T94033 CTD9M6 427880 IC50 = 4080 nM T94033 CB9VP7 432298 Ki = 2670 nM T94033 CFW9P1 441688 IC50 = 75000 nM T94033 C6VDZ3 444153 Ki = 0.071 nM T94033 CL3NE2 444469 Ki = 10 nM T94033 C3YP0R 444562 Ki = 145 nM T94033 CLV8O0 444602 IC50 = 390 nM T94033 C2DO7P 444603 Ki = 3.44 nM T94033 CZ17HE 445157 Ki = 4 nM T94033 C3R5AJ 445480 Ki > 4000 nM T94033 CRN1F6 445481 Ki > 4000 nM T94033 C2Z0XW 445482 Ki > 4000 nM T94033 CR4KE5 445844 Ki = 60000 nM T94033 CU6X2A 445847 Ki = 23000 nM T94033 CVNP24 446805 IC50 = 1500 nM T94033 C4M8WT 446979 Ki = 2460 nM T94033 CS4OB0 446982 Ki = 1610 nM T94033 C5E3YX 446984 Ki = 1420 nM T94033 C17BWY 447193 Ki = 840 nM T94033 CM3T9E 447194 Ki = 60 nM T94033 C4W7EG 447219 IC50 = 4.2 nM T94033 CD0XK3 447221 Ki = 1 nM T94033 CZC4U1 447359 Ki > 4000 nM T94033 CNO6G5 447360 Ki > 4000 nM T94033 C85OTU 447361 Ki > 3900 nM T94033 C9QXV5 447362 Ki > 4000 nM T94033 CP7V6B 447430 Ki = 0.4 nM T94033 C5UX1L 447478 Ki = 7500 nM T94033 CVND42 447482 Ki = 15000 nM T94033 C4OKV5 447486 Ki = 90000 nM T94033 CC9G5O 447490 Ki = 11000 nM T94033 CR2DX3 447496 Ki = 2300 nM T94033 COYS31 447502 Ki = 33000 nM T94033 CVI28M 447508 Ki = 180 nM T94033 CS09BE 447510 Ki = 2700 nM T94033 C87GLP 447540 Ki = 16000 nM T94033 CHV71I 447697 IC50 = 0.0017 nM T94033 C87OTC 447733 IC50 > 62000 nM T94033 CF6D4B 447734 Ki = 5580 nM T94033 CHT05K 447735 Ki = 4990 nM T94033 CK9Q4X 448061 Ki = 22000 nM T94033 C43LRO 448062 Ki = 40 nM T94033 COK45L 448065 Ki = 230 nM T94033 C5FG9U 448513 Ki = 3162277.66 nM T94033 CFMI91 448548 Ki = 13000 nM T94033 C5QKC3 448605 Ki = 940 nM T94033 CX5MS1 448610 Ki = 3200 nM T94033 C5EH8P 448675 Ki = 3 nM T94033 C02CVI 448677 Ki = 0.74 nM T94033 C4VU5J 448956 Ki = 23 nM T94033 CSL82K 449091 Ki = 1400 nM T94033 C8VB4U 480183 Ki = 10100 nM T94033 CROX25 480185 Ki = 5300 nM T94033 CGU9L8 511106 IC50 > 200000 nM T94033 CT0P5D 511111 IC50 > 200000 nM T94033 C2J3VS 576480 Ki = 100000000 nM T94033 CW02PS 603511 IC50 = 8800 nM T94033 CAO5R4 632059 IC50 >= 30000 nM T94033 COK61H 639391 Ki = 530 nM T94033 CZ8B4G 656913 Ki = 2.3 nM T94033 CP3JS0 656916 Ki = 0.0014 nM T94033 COWV76 657006 Ki = 7.7 nM T94033 C6OLN1 657007 Ki = 21 nM T94033 C53FNM 674593 IC50 = 51 nM T94033 C45NBS 674629 IC50 = 2800 nM T94033 C21HDC 674632 IC50 = 680 nM T94033 CBX3U0 674652 IC50 = 6900 nM T94033 CW5ZA1 680939 IC50 = 120 nM T94033 CG42MZ 821599 Ki = 2430000 nM T94033 CLR3H1 899247 IC50 = 4800 nM T94033 C7MYN6 1273163 IC50 = 5000 nM T94033 C5KW8I 1550286 IC50 = 89000 nM T94033 CFPA02 2392241 Ki = 290 nM T94033 CER5L6 2796875 Ki > 5000 nM T94033 C70WLF 2872455 IC50 >= 30000 nM T94033 C4S9WR 3000497 Ki = 1160 nM T94033 C4Z0XK 3010932 Ki = 279 nM T94033 CTE79D 3011892 Ki > 50000 nM T94033 C40DHV 3016780 Ki > 100000000 nM T94033 CTIR30 3081453 IC50 = 601000 nM T94033 CU43OY 3088969 Ki > 50000 nM T94033 C0K7TF 3123858 IC50 > 50000 nM T94033 C8KD9E 3162843 IC50 > 50000 nM T94033 CIK93A 3348131 Ki = 12300 nM T94033 CB58JC 3357702 Ki = 10000000 nM T94033 C4BW1J 3487462 Ki = 225 nM T94033 CK8UH3 3525149 Ki = 91 nM T94033 CZ9ST3 3564407 Ki = 158489.32 nM T94033 CA9L1G 3615188 Ki = 203 nM T94033 CQN37D 3642227 Ki = 170 nM T94033 C7ZTI9 3676069 Ki = 1995262.31 nM T94033 CFO19I 4077864 Ki = 190 nM T94033 CP4EB7 4143375 Ki = 125 nM T94033 C9FJI6 4159055 Ki = 240 nM T94033 C7XDW9 4189952 Ki = 139 nM T94033 CWKO45 4194830 Ki = 213 nM T94033 CWZY80 4231552 Ki = 212 nM T94033 CX2D9F 4348756 Ki = 227 nM T94033 CFO39X 4369278 Ki = 0.09 nM T94033 CE4V0M 4424591 Ki = 220 nM T94033 C04FRG 4454738 Ki = 225 nM T94033 C7WO3C 4607840 Ki = 123 nM T94033 C8EK6S 4620241 Ki = 1584893.19 nM T94033 CCT23L 4634566 Ki = 4000 nM T94033 CT8JE1 4655928 Ki > 5000 nM T94033 CAE8O5 4670471 Ki = 240 nM T94033 C9SJZ7 5048318 Ki = 1584893.19 nM T94033 C25HKV 5058442 Ki = 130 nM T94033 C7XQ0G 5073138 Ki = 219 nM T94033 CEBR63 5074355 Ki = 146 nM T94033 CV95FQ 5108695 Ki = 794328.23 nM T94033 CV7AX9 5172545 Ki = 431000 nM T94033 C1I9XL 5183332 Ki = 129 nM T94033 CG7BH6 5221300 Ki = 1000000 nM T94033 CPZ6A3 5287506 Ki = 35 nM T94033 CWS92L 5287523 IC50 = 1000 nM T94033 C48TEQ 5287836 Ki = 1260 nM T94033 C51HAG 5287925 IC50 = 49 nM T94033 C2L7EJ 5287991 Ki = 1 nM T94033 C1YGX2 5289320 Ki = 12300 nM T94033 C8I0VG 5289529 Ki = 7100 nM T94033 CQ26VM 5289531 Ki = 3300 nM T94033 CNB7Q3 5328796 Ki = 102000 nM T94033 C1B9GP 5400404 IC50 > 50000 nM T94033 C6F8LD 5478933 Ki = 2.01 nM T94033 C0CV5L 5496928 IC50 > 100000 nM T94033 CAW1P7 5497056 Ki ~ 2900 nM T94033 CW59HK 5760260 Ki = 165000 nM T94033 C7SYK9 6102731 IC50 = 24000 nM T94033 C3IPA1 6367052 Ki = 300 nM T94033 CEB3W0 6426822 Ki = 0.35 nM T94033 CYJ4I8 6476665 IC50 > 200000 nM T94033 C2ZRF5 6540265 IC50 = 420 nM T94033 CN57IY 6540268 IC50 = 20 nM T94033 C4W9BX 6852123 Ki = 1900 nM T94033 CFJ8Q1 6852188 IC50 = 1 nM T94033 CN2B6S 6852211 Ki = 5000 nM T94033 C49IOZ 6857707 Ki = 60000 nM T94033 C8OE6S 6913584 IC50 = 3660 nM T94033 CHW7K8 6914575 IC50 = 3.2 nM T94033 CM8R6E 6914706 IC50 > 1200000 nM T94033 CF4TK5 8967105 IC50 >= 30000 nM T94033 CNZA87 9112697 IC50 > 200000 nM T94033 CG9B5V 9543484 IC50 = 3.7 nM T94033 CWR2K4 9543485 IC50 = 220 nM T94033 C4B1EW 9543486 IC50 = 100000 nM T94033 CXTU39 9543487 IC50 = 12000 nM T94033 CX34ZD 9549214 Ki = 780 nM T94033 CP3QT1 9560223 Ki = 68000 nM T94033 C7XL2M 9573034 Ki = 786000 nM T94033 CK64FD 9794516 IC50 = 130 nM T94033 C6JDM9 9799627 Ki = 6440 nM T94033 CVFE34 9800775 IC50 > 10000 nM T94033 C92QSE 9801235 IC50 > 100000 nM T94033 C2FHU7 9801905 IC50 = 19 nM T94033 CL1R0T 9801948 Ki = 18 nM T94033 C6ZD2L 9802069 Ki = 11 nM T94033 C40LRN 9802229 Ki = 7.4 nM T94033 CYL75R 9802758 Ki = 11 nM T94033 C3FS0U 9802858 Ki = 19 nM T94033 C4VX9Y 9803558 IC50 > 10000 nM T94033 CS91FJ 9803642 Ki = 8.3 nM T94033 CTA52P 9803848 Ki = 35 nM T94033 C07DSH 9804052 Ki = 1.6 nM T94033 C8QGS1 9804434 Ki > 21000 nM T94033 CDN8P2 9804727 Ki = 170 nM T94033 C1FIN6 9804775 IC50 > 130 nM T94033 CHJB86 9805409 Ki = 2.4 nM T94033 C4OTK6 9805415 IC50 > 10000 nM T94033 CAKN38 9805632 Ki > 21000 nM T94033 C6JIT7 9806444 IC50 > 11000 nM T94033 CBKL18 9806644 IC50 > 10000 nM T94033 C2WHZ0 9806941 IC50 = 120 nM T94033 CW3NK6 9806974 Ki = 11000 nM T94033 C6F3XK 9807686 Ki > 1500000 nM T94033 C6JY9R 9807737 Ki = 0.004 nM T94033 CAG59M 9808035 Ki = 1400 nM T94033 CTS98Y 9808170 Ki = 15000 nM T94033 CH9IE6 9808346 Ki = 2540 nM T94033 CZS3H5 9808724 Ki > 6300 nM T94033 C2AXV0 9809479 Ki = 1600 nM T94033 C8UX0O 9810198 Ki > 1000000 nM T94033 C60AVD 9812184 Ki = 14000 nM T94033 CLTO67 9821317 IC50 > 100000 nM T94033 C4KEZ2 9821506 Ki = 300 nM T94033 CKN89B 9822176 Ki > 30000 nM T94033 CD5M9P 9823195 Ki = 140 nM T94033 CJ2G7A 9823668 IC50 > 10000 nM T94033 CX6DA7 9823789 Ki = 9900 nM T94033 CH5F9G 9823849 Ki = 44 nM T94033 CXT07H 9824011 IC50 = 14000 nM T94033 CD3AP6 9824122 Ki > 21000 nM T94033 C0QH1L 9824657 Ki = 2.3 nM T94033 CZ64PW 9824925 Ki > 21000 nM T94033 C9RB6Q 9825365 IC50 = 2.7 nM T94033 CTG89N 9825830 Ki = 771 nM T94033 C08XFQ 9825841 Ki = 0.37 nM T94033 CPB20R 9826345 Ki = 1000 nM T94033 CS1DL7 9826716 IC50 > 11000 nM T94033 CB82VS 9827306 IC50 > 11000 nM T94033 CGN48U 9827867 IC50 = 196 nM T94033 CE0HD3 9828470 Ki = 280 nM T94033 COW7Q3 9829120 IC50 = 4800 nM T94033 CP2X5B 9829453 Ki = 8000 nM T94033 C8RV5E 9830070 Ki > 21000 nM T94033 C4F8CN 9830285 IC50 < 40 nM T94033 CGNB60 9830581 IC50 = 3600 nM T94033 C4T5BQ 9830932 Ki = 2000 nM T94033 C71OHU 9831158 Ki = 0.78 nM T94033 C6W8QC 9831694 IC50 = 80 nM T94033 C1WK3X 9838954 Ki = 700 nM T94033 CH38SL 9840270 Ki = 710000 nM T94033 C58QBT 9842536 Ki = 18 nM T94033 C14HZE 9842688 Ki = 390 nM T94033 CVO5R3 9842851 IC50 > 10000 nM T94033 C7UOA2 9844807 Ki = 270 nM T94033 CC4Y8V 9845104 Ki = 6500 nM T94033 C6VAG8 9845526 IC50 = 8 nM T94033 C2TA1I 9845742 IC50 = 950 nM T94033 CM8Y9G 9846259 IC50 > 100000 nM T94033 CY7FU4 9846410 Ki = 2.1 nM T94033 C8I4LS 9846496 Ki > 21000 nM T94033 CE5H2V 9846562 Ki = 7 nM T94033 CM0OU9 9847373 IC50 = 12.4 nM T94033 C69RDJ 9847494 Ki > 10000 nM T94033 CU2H1W 9848037 IC50 > 10000 nM T94033 C5Z2RH 9848091 IC50 > 11000 nM T94033 CX8NG2 9848165 Ki = 0.26 nM T94033 CX25MR 9848465 Ki = 1900 nM T94033 CW3EC6 9848592 Ki = 43 nM T94033 CCL5G3 9848846 IC50 > 10000 nM T94033 CED43L 9850077 IC50 = 21 nM T94033 CE0K4C 9850350 IC50 = 11 nM T94033 CS9HQ0 9850467 Ki = 0.85 nM T94033 CT7S2K 9850497 Ki = 0.003 nM T94033 C3F0CS 9851859 Ki = 147 nM T94033 C75JUE 9853816 IC50 = 2320 nM T94033 CP8CY7 9859977 IC50 > 200000 nM T94033 CY7B8Q 9860803 Ki = 4700 nM T94033 CB86RC 9864323 Ki = 110 nM T94033 CF74PR 9864759 IC50 > 10000 nM T94033 CSH3K5 9865994 Ki = 2.3 nM T94033 C8T6JE 9867609 Ki = 1.2 nM T94033 CY6EA8 9868194 Ki = 10 nM T94033 CYDE28 9868624 IC50 = 1.68 nM T94033 C89JRZ 9868633 Ki = 0.82 nM T94033 CQ5J9K 9868873 Ki = 540 nM T94033 CL6QS0 9868922 Ki = 100 nM T94033 CDVE40 9869375 IC50 > 10000 nM T94033 C3P1EU 9869891 Ki = 0.76 nM T94033 C38BTY 9870834 Ki = 12000 nM T94033 CZ9LR2 9870910 Ki = 48 nM T94033 C1AW6N 9870947 Ki = 53000 nM T94033 CIL85V 9871029 IC50 > 11000 nM T94033 C8ZXJ5 9871065 Ki = 2.4 nM T94033 C9UB6X 9871197 Ki > 21000 nM T94033 CIZ61P 9872423 Ki = 140 nM T94033 C8O3SW 9872549 Ki = 0.04 nM T94033 C6ZB3K 9872552 IC50 > 11000 nM T94033 C87SWZ 9872983 Ki > 1000000 nM T94033 CG0L6A 9873029 IC50 = 8640 nM T94033 C5LV1Z 9873979 Ki = 22 nM T94033 CJ1XE3 9874681 Ki = 1.2 nM T94033 CA9Z4S 9875345 Ki = 435000 nM T94033 CPU3D1 9881263 IC50 = 129000 nM T94033 CS78YB 9882885 IC50 > 200000 nM T94033 C2F5NS 9884570 Ki = 7500 nM T94033 CQP0V2 9886960 Ki = 380 nM T94033 CJT9X7 9887558 Ki = 2000 nM T94033 CAW39H 9888145 Ki = 1.6 nM T94033 C2IR9Z 9889864 IC50 = 1900 nM T94033 CYKX52 9889871 Ki = 0.75 nM T94033 C6A4TL 9890540 Ki > 21000 nM T94033 C17NPU 9890541 IC50 = 0.505 nM T94033 C3Y8AL 9890583 Ki = 6.8 nM T94033 C7ALY1 9890731 Ki = 6.7 nM T94033 C46LWX 9890816 Ki = 3.1 nM T94033 CP4B3U 9890882 IC50 = 5.4 nM T94033 C0RO1Q 9891135 Ki = 0.49 nM T94033 CO4QD2 9891154 Ki = 4000 nM T94033 CO4KT2 9891302 Ki = 0.53 nM T94033 C7E1IV 9891337 IC50 = 0.71 nM T94033 CT6W0R 9891759 Ki > 3500 nM T94033 CD13TH 9891795 IC50 > 10000 nM T94033 C1M2PU 9892103 IC50 > 11000 nM T94033 C8UV6Y 9892106 Ki = 6500 nM T94033 C7I5RG 9892392 Ki = 19000 nM T94033 CXY68Z 9893122 IC50 > 10000 nM T94033 CNJ0W1 9893177 IC50 = 1 nM T94033 C5IG2W 9893544 Ki = 1500 nM T94033 CW3J0F 9893616 IC50 = 58 nM T94033 CV3F0R 9893703 Ki = 1.8 nM T94033 CK74IX 9894066 Ki = 0.65 nM T94033 C4DHN5 9894203 Ki > 21000 nM T94033 CB4O8L 9894223 Ki > 21000 nM T94033 C13KVD 9894553 Ki > 6300 nM T94033 C9SJ3T 9894908 IC50 = 18 nM T94033 CKDP84 9895193 Ki = 490 nM T94033 C6PSQ7 9896889 Ki = 138000 nM T94033 CZY9L0 9905436 IC50 = 134000 nM T94033 C0SP6Q 9906596 Ki = 1200 nM T94033 C2HN7L 9907201 Ki = 1100 nM T94033 C85SEZ 9908687 IC50 > 10000 nM T94033 CMG5R2 9909967 Ki = 460 nM T94033 CMC95R 9910164 IC50 = 1.5 nM T94033 CAP0O8 9910540 Ki = 2900 nM T94033 CQ7PT5 9910790 Ki = 1.7 nM T94033 CD5LQ0 9910982 Ki = 4.6 nM T94033 CAWD59 9911275 IC50 > 100000 nM T94033 C5HS9Y 9911866 Ki = 0.5 nM T94033 C21RUG 9911960 Ki = 0.4 nM T94033 CL0K6H 9912101 Ki = 3.9 nM T94033 CO52XJ 9912171 Ki = 1.1 nM T94033 CS6QF5 9912191 Ki > 21000 nM T94033 CNB6I1 9912441 Ki = 7.3 nM T94033 C0LKE7 9912771 Ki > 100000 nM T94033 C8GJF3 9913055 IC50 = 0.71 nM T94033 CNT57V 9913233 Ki = 2.9 nM T94033 CXF4P3 9913838 Ki = 2.4 nM T94033 C2MR5K 9914088 IC50 = 49 nM T94033 C1C3VT 9914538 IC50 > 11000 nM T94033 CCB64X 9914780 Ki = 1.1 nM T94033 CC0D5H 9915041 Ki = 3600 nM T94033 CPZ50Y 9915193 Ki = 300 nM T94033 CVND52 9915545 Ki = 33200 nM T94033 C2GWH3 9916339 Ki > 21000 nM T94033 CHG59Y 9916885 Ki > 1500000 nM T94033 CK2H1C 9917705 Ki = 400 nM T94033 CG36KH 9919038 IC50 = 570 nM T94033 CFO1K9 9922130 Ki > 1000000 nM T94033 CLZ53G 9922131 Ki = 200000 nM T94033 CAP64B 9929157 Ki = 3100 nM T94033 C2TO4N 9931543 Ki > 6600 nM T94033 C7ZJ5X 9931673 Ki = 830 nM T94033 CS7LF5 9931725 Ki = 11 nM T94033 CRD3A7 9931726 Ki = 11 nM T94033 C9I2ES 9931785 IC50 = 3 nM T94033 CE6O2X 9932142 IC50 = 25.12 nM T94033 C4EJB2 9933009 IC50 = 19000 nM T94033 C85LIU 9934003 Ki = 2000 nM T94033 CS9Y5I 9934133 IC50 > 10000 nM T94033 CLT7P8 9934591 IC50 = 882 nM T94033 CI86NB 9934869 IC50 = 300 nM T94033 C38QWF 9935364 Ki = 1250 nM T94033 CG3B1P 9935390 Ki = 120 nM T94033 CM1S3V 9935481 Ki = 24 nM T94033 C1XT2Y 9935746 Ki = 6200 nM T94033 CL2NV0 9935925 IC50 > 870 nM T94033 C5KS0R 9936020 IC50 > 11000 nM T94033 CKLJ26 9936190 IC50 > 100000 nM T94033 C49DRC 9936691 IC50 > 11000 nM T94033 CR3Z9T 9936843 Ki = 2.8 nM T94033 CL0U1E 9936850 IC50 = 503 nM T94033 C41OYV 9936939 Ki = 2.4 nM T94033 CG96QC 9936983 Ki = 2400 nM T94033 COA4R0 9937032 Ki = 8900 nM T94033 CF3VC7 9937307 Ki = 0.31 nM T94033 CC9QH7 9937406 Ki = 0.65 nM T94033 C8F5CW 9937921 Ki = 6000 nM T94033 C8LR4T 9938917 Ki = 1100 nM T94033 CDT95S 9939426 Ki = 500 nM T94033 C1RHT8 9949886 Ki = 1100 nM T94033 CD27EJ 9951054 IC50 > 10000 nM T94033 CP06LN 9953722 Ki = 20 nM T94033 COR74I 9954289 Ki = 2.8 nM T94033 CWNA41 9954607 Ki = 4.5 nM T94033 C4NJU3 9954757 Ki = 12 nM T94033 CD7ZO5 9954791 Ki = 0.04 nM T94033 C0R4GE 9954812 IC50 = 321000 nM T94033 CX85LD 9954980 Ki = 7660 nM T94033 CP7A2W 9955292 Ki > 21000 nM T94033 CSI62L 9955475 IC50 > 10000 nM T94033 C3EPC4 9955758 Ki = 11.9 nM T94033 CV96ZD 9955999 Ki > 21000 nM T94033 C58QTM 9956404 Ki = 15400 nM T94033 CY5OI8 9956416 IC50 = 22000 nM T94033 CM7IF6 9956559 Ki = 0.5 nM T94033 C8Y4EG 9956632 Ki = 1600 nM T94033 C8CLF7 9956947 Ki = 0.85 nM T94033 CI84CP 9957386 Ki = 600 nM T94033 CN36AS 9957822 Ki = 3800 nM T94033 CE39JM 9958168 Ki = 5 nM T94033 C5CRQ2 9958229 Ki = 0.05 nM T94033 C3WAS5 9958320 Ki = 0.09 nM T94033 C9AW3Q 9958913 Ki = 0.6 nM T94033 CJ0E7R 9959071 Ki = 0.5 nM T94033 CLW0D4 9959111 IC50 = 8 nM T94033 C2Y0QV 9959268 IC50 > 10000 nM T94033 C1BSX7 9959541 Ki = 0.65 nM T94033 CBC2K3 9959749 IC50 > 11000 nM T94033 C0C1FQ 9959919 Ki = 800 nM T94033 C5MIF2 9960017 Ki = 39 nM T94033 COMH01 9961613 Ki = 26000 nM T94033 C8MP2G 9962253 Ki = 15000 nM T94033 C2CE1A 9962331 Ki > 50000 nM T94033 C0TV8Q 9962561 Ki = 57 nM T94033 C3HI6E 9972080 IC50 = 48990 nM T94033 CTMU52 9978512 IC50 > 1600000 nM T94033 C3S7IV 9979724 Ki = 1164 nM T94033 CV81FG 9980363 IC50 = 15000 nM T94033 C38MBH 9981197 Ki = 1550 nM T94033 C4CH0E 9981449 Ki = 4700 nM T94033 C1O6WC 9981956 Ki = 1200 nM T94033 C6XM2Z 9982428 Ki = 7400 nM T94033 CK6XE9 9982431 IC50 > 30000 nM T94033 CY3Z7I 9982644 IC50 > 10000 nM T94033 C5SA7F 9983043 IC50 = 7.95 nM T94033 C5UGC0 9983309 Ki = 48 nM T94033 CKEB95 9984267 IC50 = 13 nM T94033 CUE8L0 9984551 Ki = 100 nM T94033 CZ3U8E 9984568 Ki = 0.4 nM T94033 CD6Y1S 9985229 Ki = 26 nM T94033 CZ6TD1 9985759 Ki = 5000 nM T94033 CZQ7B4 9986265 Ki = 3.1 nM T94033 CC07LB 9987016 Ki = 0.07 nM T94033 CKP2Z7 9987204 Ki = 111 nM T94033 CKIP10 9987251 IC50 = 30000 nM T94033 CEC95B 9997816 Ki = 550 nM T94033 C25AEU 9999606 Ki = 180 nM T94033 CE75GM 10000477 IC50 = 4000 nM T94033 CO29YH 10001054 Ki = 11 nM T94033 C1FVM2 10001731 IC50 = 870 nM T94033 CJ0Q2S 10002821 Ki = 2.3 nM T94033 CVQN23 10003356 Ki = 1.2 nM T94033 C56FZK 10003877 IC50 > 10000 nM T94033 C4KCS7 10004019 Ki = 1200 nM T94033 CU9QI6 10004529 Ki = 300 nM T94033 C9O5SJ 10004800 Ki = 0.31 nM T94033 C9ZM4S 10005728 Ki = 958 nM T94033 C8I7YZ 10006319 IC50 = 89 nM T94033 CZJ38W 10006399 IC50 = 28.8 nM T94033 CBPE30 10006490 Ki = 10.9 nM T94033 CC3RI8 10006831 Ki = 0.4 nM T94033 C08RZY 10007252 Ki = 660 nM T94033 CAW18J 10007800 IC50 = 80000 nM T94033 CFQV59 10007890 IC50 > 10000 nM T94033 CTMQ73 10008817 IC50 = 72000 nM T94033 CWMC62 10009177 IC50 < 1 nM T94033 C7LWC0 10009777 IC50 = 9 ug.mL-1 T94033 C98OVC 10021822 Ki = 1300 nM T94033 C0A6SH 10022303 Ki = 180 nM T94033 CB1SY8 10023491 IC50 > 1000000 nM T94033 CH7AS9 10023890 Ki = 25 nM T94033 C05LTI 10024002 IC50 = 130 nM T94033 C8ME3O 10024183 Ki = 1.7 nM T94033 CDF1Q4 10025885 Ki = 1.5 nM T94033 CBL8D4 10026170 Ki = 0.42 nM T94033 CHP0G5 10027333 Ki = 0.04 nM T94033 CF1V4K 10027758 Ki > 4000 nM T94033 CW5JH1 10028252 Ki = 170 nM T94033 CEH0M2 10028749 Ki = 6.6 nM T94033 C3SU6O 10028986 Ki = 970 nM T94033 CX4TI5 10029172 Ki = 3000 nM T94033 C3E4DR 10029213 IC50 = 85 nM T94033 C4PFW9 10029239 Ki = 4600 nM T94033 CI2O5B 10029343 IC50 = 5400 nM T94033 CB4Y7M 10030046 IC50 = 1000 nM T94033 CYF86J 10030346 Ki = 11 nM T94033 C0ZV2H 10030708 Ki = 13 nM T94033 CJPR86 10031628 Ki = 0.68 nM T94033 C8KIA9 10037020 IC50 = 6 nM T94033 CUG6R3 10037159 Ki = 720 nM T94033 CSX68Z 10043156 IC50 > 10000 nM T94033 C6XT4N 10043206 Ki = 10 nM T94033 CU7A2O 10047384 Ki = 16000 nM T94033 CC9Y8U 10047767 Ki = 9 nM T94033 CK4W6M 10047815 IC50 = 20000 nM T94033 CAO7B5 10048535 Ki = 3.4 nM T94033 C9R8YW 10048823 Ki = 4.6 nM T94033 C8TM7V 10048854 Ki = 600 nM T94033 C8FKM2 10049151 IC50 > 10000 nM T94033 C80QYS 10051154 Ki = 120 nM T94033 C08PUS 10051441 IC50 = 12 nM T94033 CVY28G 10051489 Ki = 0.16 nM T94033 C29DTM 10051582 Ki = 180 nM T94033 CU9I7D 10051599 Ki = 1500 nM T94033 CHZL08 10051960 Ki = 2400 nM T94033 C3QP6V 10052373 Ki = 4.6 nM T94033 CFCT67 10053115 Ki = 330 nM T94033 CDE42G 10053298 Ki = 11000 nM T94033 C6R5AP 10053447 Ki = 4.8 nM T94033 C9KC6Q 10053945 IC50 = 110 nM T94033 CXZ2V3 10054210 Ki = 200 nM T94033 CHAY26 10055165 Ki = 63 nM T94033 C8YHP3 10055497 Ki = 111000 nM T94033 CL2J6U 10060627 Ki = 260 nM T94033 C1OI8R 10066101 Ki = 2200 nM T94033 C6F4SZ 10067786 Ki = 1.7 nM T94033 CBV7N2 10070407 IC50 = 25 nM T94033 CPR1C7 10070588 Ki = 6.6 nM T94033 CW28HS 10071127 Ki = 620 nM T94033 CRID91 10071900 IC50 > 333000 nM T94033 CI2KG6 10072299 IC50 > 30000 nM T94033 CPR8A3 10072533 IC50 = 0.9 nM T94033 CP65QI 10073006 Ki = 300 nM T94033 C7TU4O 10073666 Ki > 5000 nM T94033 CB04YW 10073864 IC50 = 8000 nM T94033 CP5BK0 10074165 Ki = 0.001 nM T94033 CF4R2W 10074230 IC50 = 16 nM T94033 CUOC38 10074752 Ki = 0.52 nM T94033 CO0N7Q 10074781 Ki = 1890 nM T94033 CAT42M 10074892 Ki = 100 nM T94033 C9ZCS2 10074922 IC50 = 30 nM T94033 CF0R6D 10074927 IC50 = 0.67 nM T94033 CD5AT6 10075317 Ki = 0.4 nM T94033 C61CAI 10075751 Ki = 18 nM T94033 CWM85P 10076656 IC50 = 1410 nM T94033 C4B7NV 10077222 IC50 > 200000 nM T94033 CD0VO9 10078364 IC50 = 4000 nM T94033 C7CW1P 10080504 IC50 = 5600 nM T94033 CR0ZL7 10091675 IC50 = 18 nM T94033 CP38MH 10091962 IC50 = 230000 nM T94033 CVC9O4 10092169 IC50 = 890 nM T94033 CZM79H 10093390 Ki = 260 nM T94033 C1HIC3 10093417 Ki = 1.2 nM T94033 CEN06H 10093642 IC50 = 35000 nM T94033 C4P3ZO 10093667 IC50 > 10000 nM T94033 C3TDM1 10094168 Ki = 3250 nM T94033 C2VT9U 10094219 Ki > 4000 nM T94033 CZH3W7 10094378 Ki = 11 nM T94033 C0FS4U 10094458 IC50 > 400000 nM T94033 CMHD92 10094532 IC50 > 10000 nM T94033 CRXD40 10095024 Ki = 220 nM T94033 C6PVA7 10095315 IC50 > 10000 nM T94033 C3TWI1 10095455 IC50 = 20 nM T94033 C3OG5U 10095865 Ki = 2 nM T94033 C0JE3C 10096795 IC50 > 10000 nM T94033 CW6LB3 10097039 Ki = 0.046 nM T94033 CC5G8U 10097473 Ki = 14 nM T94033 C3IRT4 10098156 Ki > 13000 nM T94033 CRS8D1 10098302 Ki = 0.07 nM T94033 CX8A6G 10099038 Ki > 13000 nM T94033 CO8G7N 10099218 IC50 = 1000 nM T94033 CV6NQ3 10099674 Ki > 13000 nM T94033 C02SZJ 10100610 Ki = 70 nM T94033 CQB1V2 10101474 IC50 = 0.04 ug.mL-1 T94033 CMOE48 10113121 Ki = 0.12 nM T94033 CK01GN 10114268 Ki = 157.9 nM T94033 CM5BQ6 10114365 Ki = 47 nM T94033 COH4E2 10115868 Ki = 16 nM T94033 C1TO0F 10115923 Ki = 2.7 nM T94033 C0AFU1 10116445 Ki > 4000 nM T94033 CW4RZ5 10116936 IC50 > 450 nM T94033 C1VT4F 10117027 Ki = 7500 nM T94033 C9V2WC 10117161 IC50 > 10000 nM T94033 CW1AG0 10117424 Ki = 1.4 nM T94033 CXCR46 10117543 Ki = 470 nM T94033 C1XZ8N 10117556 IC50 > 100000 nM T94033 CH3L1P 10117895 Ki = 0.096 nM T94033 CL4Q3M 10118619 Ki = 1.2 nM T94033 C7P6IV 10119176 Ki = 0.017 nM T94033 C9PG6D 10119254 Ki = 900 nM T94033 CE2DI8 10119483 Ki = 0.0014 nM T94033 CX9VL6 10119957 Ki = 0.003 nM T94033 CV5E4L 10121049 Ki > 35100 nM T94033 C4TB7E 10121121 Ki = 4900 nM T94033 CR03NV 10131788 Ki > 1000000 nM T94033 C3EFH5 10136204 Ki = 6.7 nM T94033 CVA35H 10140425 Ki = 5.9 nM T94033 CS2G4T 10140847 Ki = 290 nM T94033 CMFW67 10140911 Ki = 34 nM T94033 C67VZS 10141105 IC50 = 877 nM T94033 C9CBP0 10141313 Ki = 7.3 nM T94033 CWF4I3 10141502 Ki = 12000 nM T94033 CN2WO7 10141594 Ki = 200 nM T94033 C1Q3KU 10141691 Ki = 900 nM T94033 C31QAL 10143532 Ki = 300 nM T94033 C7L5IJ 10157296 Ki = 130 nM T94033 C4K3WG 10162441 Ki = 0.1 nM T94033 CT65YJ 10162799 Ki = 4 nM T94033 CBHY78 10163266 Ki = 6 nM T94033 CF82TK 10163421 Ki = 20000 nM T94033 C75ADN 10164065 Ki = 8000 nM T94033 C9B2CI 10164798 Ki = 0.085 nM T94033 CM6PS4 10165173 Ki = 4200 nM T94033 C6Y9DT 10165269 Ki = 0.03 nM T94033 C1QBH5 10165288 Ki = 0.018 nM T94033 CDRK68 10165573 Ki < 0.01 nM T94033 C5WB4J 10165649 Ki = 690 nM T94033 C7G4JC 10166616 Ki > 35100 nM T94033 CEPJ05 10166622 Ki = 3330 nM T94033 C5I0YH 10168444 Ki > 100000 nM T94033 CG37YX 10181104 IC50 > 30000 nM T94033 CF4S8B 10183471 Ki = 1100 nM T94033 CT31ZH 10183608 Ki = 5.3 nM T94033 C20EJH 10183697 Ki = 281 nM T94033 CM0X5B 10184785 Ki > 21000 nM T94033 C7PC2K 10185292 IC50 > 170 nM T94033 C93EKT 10185327 Ki = 1.6 nM T94033 CFN3T0 10185355 Ki = 6.3 nM T94033 CFIH78 10185526 IC50 = 21700 nM T94033 CU24HL 10186048 Ki > 21000 nM T94033 C1DN4F 10187311 Ki = 360 nM T94033 CD9JP8 10188053 Ki = 0.008 nM T94033 CAK19V 10188881 Ki = 4500 nM T94033 CZ9KS7 10188952 Ki > 21000 nM T94033 CF2E6U 10198683 IC50 = 14400 nM T94033 CHY62J 10203373 Ki > 21000 nM T94033 CMT1R3 10204622 Ki = 85.2 nM T94033 CO51ZR 10205659 IC50 > 10000 nM T94033 CY23WJ 10205851 Ki = 3.3 nM T94033 C2CWI1 10206231 Ki = 1.1 nM T94033 C27JIT 10207236 Ki = 0.45 nM T94033 CV2F6G 10207343 Ki = 0.14 nM T94033 CO4QT2 10207346 IC50 > 10000 nM T94033 CGP08H 10207789 Ki = 3.1 nM T94033 CW62PU 10207853 Ki = 900 nM T94033 C4YET3 10208026 Ki = 0.21 nM T94033 CT0S2D 10208075 Ki = 0.013 nM T94033 CDCZ31 10208076 Ki = 0.84 nM T94033 CI6VM2 10208564 Ki = 0.013 nM T94033 C01QTR 10209142 Ki = 5380 nM T94033 CP69QR 10212999 IC50 > 10000 nM T94033 CJRS38 10217801 Ki = 3500 nM T94033 CQU78Y 10222156 Ki = 290 nM T94033 C8V1AY 10225952 Ki = 120 nM T94033 CR6K3D 10226645 Ki = 10.3 nM T94033 C6HAC0 10227428 Ki = 1500 nM T94033 CT18AE 10227443 Ki ~ 4000 nM T94033 CIAX57 10228506 Ki = 590 nM T94033 CSR74M 10228660 IC50 > 100000 nM T94033 CN1PX4 10228720 Ki > 21000 nM T94033 CIGQ87 10228750 Ki = 6.9 nM T94033 CEP76D 10228869 Ki = 940 nM T94033 CY41MS 10228870 Ki = 0.033 nM T94033 C98FSX 10230007 Ki = 610 nM T94033 C4RSF3 10230057 Ki = 0.16 nM T94033 CMU21W 10231661 Ki = 530 nM T94033 C7G5XE 10239342 Ki = 1700 nM T94033 CF4ND2 10247830 Ki = 3000 nM T94033 C2XHG8 10248900 Ki > 29000 nM T94033 CYJ7C6 10249621 IC50 = 94 nM T94033 C9QML3 10250104 Ki = 3300 nM T94033 C7RVY1 10253674 Ki = 3800 nM T94033 CXM94D 10255216 IC50 = 56.23 nM T94033 C4Z1LU 10255253 Ki > 4000 nM T94033 C53DHK 10255441 Ki = 3950 nM T94033 C71RTC 10255760 IC50 > 10000 nM T94033 CX0MW3 10255784 IC50 = 100000 nM T94033 C9IAO4 10256095 IC50 = 1250 nM T94033 CS4F5P 10256448 IC50 = 190 nM T94033 CIA4E1 10256748 Ki = 0.6 nM T94033 CD6V5R 10256934 IC50 = 1350 nM T94033 C4WV1A 10257345 IC50 > 2500 nM T94033 CFBN38 10257580 IC50 = 4700 nM T94033 C2F4TQ 10259285 Ki = 20800 nM T94033 CSX60M 10264543 Ki = 37870 nM T94033 C3X6SG 10273187 Ki = 2.1 nM T94033 C9E8OU 10273521 Ki = 0.57 nM T94033 CQ9ZO1 10275412 Ki > 15000 nM T94033 CNE1I4 10277604 Ki = 7.2 nM T94033 CONF80 10277810 Ki = 3.6 nM T94033 C0J1TD 10278414 Ki = 170 nM T94033 C50WLH 10278497 IC50 > 10000 nM T94033 C3M5KS 10279315 Ki = 0.0034 nM T94033 CD1BR9 10280794 Ki = 0.015 nM T94033 CB1S5P 10281431 Ki > 35100 nM T94033 CXL1S0 10289409 Ki = 157 nM T94033 CZM97W 10293977 Ki = 69000 nM T94033 C5EDW1 10294146 Ki = 360 nM T94033 C0T3CN 10296435 IC50 > 100000 nM T94033 CP2V3F 10297781 IC50 = 1400 nM T94033 CV10CU 10297977 IC50 > 10000 nM T94033 CM62FC 10298615 IC50 > 10000 nM T94033 C1AP6H 10298858 IC50 > 10000 nM T94033 C79BFH 10298942 Ki > 15000 nM T94033 CPX8N9 10299701 Ki = 4400 nM T94033 CDP9R7 10299889 Ki > 21000 nM T94033 CLJ02I 10300491 Ki = 3300 nM T94033 C4DSV3 10300585 Ki = 7.2 nM T94033 CN2OL6 10300646 Ki = 3.5 nM T94033 CA5L9Q 10300692 Ki = 0.66 nM T94033 CEW97F 10301102 Ki = 9 nM T94033 CU59LR 10301422 Ki = 5.8 nM T94033 C8XLH9 10302418 Ki = 27300 nM T94033 C6WH5B 10303315 Ki = 0.01 nM T94033 CGTF74 10303947 Ki > 35100 nM T94033 C17RDU 10304095 Ki = 31 nM T94033 C8PA9J 10310498 Ki = 10000 nM T94033 CN8FL2 10315612 Ki = 4900 nM T94033 CMR75W 10318568 IC50 > 100000 nM T94033 C25XSY 10318999 IC50 > 100000 nM T94033 CUN7Z6 10321113 Ki = 1.5 nM T94033 COU98F 10321592 Ki = 6 nM T94033 C8Y4EJ 10322243 Ki = 360 nM T94033 CQXH16 10323441 Ki = 32 nM T94033 CMR6Y8 10323469 IC50 = 6300 nM T94033 C8SQ1N 10324263 Ki = 7800 nM T94033 CX9J5U 10324635 Ki = 0.14 nM T94033 CA1PG7 10324778 Ki = 9 nM T94033 CT0FX4 10325259 Ki > 13000 nM T94033 CSJ12N 10325266 Ki = 38 nM T94033 C56PEV 10325271 IC50 = 1.5 nM T94033 C90OGN 10325899 IC50 = 154000 nM T94033 C41ZLB 10326602 IC50 > 2500 nM T94033 CC8QH1 10326719 Ki = 10 nM T94033 C53QGN 10339033 Ki = 150 nM T94033 CN5R3I 10340020 Ki = 3.1 nM T94033 CZMH83 10340538 IC50 = 9000 nM T94033 C92ULP 10340574 Ki = 3.7 nM T94033 C4YR1M 10342318 Ki = 5200 nM T94033 C8ZEL7 10342377 IC50 > 1000000 nM T94033 CP64HV 10342843 Ki = 2 nM T94033 CV8J6G 10343097 Ki = 2390 nM T94033 CFL57Y 10343633 Ki = 2100 nM T94033 CK9J7X 10343728 Ki = 17 nM T94033 C4I7DQ 10345176 Ki = 32 nM T94033 C8FO7Q 10345230 Ki = 191 nM T94033 CES6C2 10345244 Ki = 7800 nM T94033 CE90ON 10345251 Ki = 3 nM T94033 CF9Q3K 10345602 Ki = 5 nM T94033 CH0RW2 10346646 IC50 > 10000 nM T94033 C9H8XN 10347184 IC50 = 57100 nM T94033 CUX6P9 10347185 IC50 = 2500 nM T94033 C4KER5 10347610 IC50 > 10000 nM T94033 COP0E1 10347939 Ki = 2.6 nM T94033 C9LB3S 10347951 IC50 = 330000 nM T94033 CK87NT 10348221 Ki = 3.5 nM T94033 C5RK3D 10348577 Ki = 0.71 nM T94033 CFUM15 10348619 Ki = 330 nM T94033 CHC08V 10349473 Ki = 3.5 nM T94033 CL09QG 10349678 IC50 = 100000 nM T94033 C83DLG 10361934 Ki = 430 nM T94033 C6MB8U 10362976 IC50 = 980 nM T94033 CL07UC 10364218 Ki = 16400 nM T94033 CW29YO 10365461 IC50 > 600000 nM T94033 CS3U1O 10365507 Ki = 10 nM T94033 CH0V8B 10366070 Ki = 17800 nM T94033 C0ODK9 10366157 IC50 > 10000 nM T94033 C0XW1E 10366176 IC50 = 22000 nM T94033 C2E4TL 10366902 IC50 = 6.2 nM T94033 C10ISY 10367012 Ki = 0.056 nM T94033 C4JC7H 10367232 IC50 > 300000 nM T94033 C1D4YB 10367245 Ki = 2.17 nM T94033 CJ0O5P 10367277 IC50 > 33000 nM T94033 CIQ63E 10367299 IC50 > 10000 nM T94033 CG98CM 10367552 Ki = 2100 nM T94033 CM2YJ6 10367719 Ki = 0.6 nM T94033 C5T6DO 10367956 Ki = 0.04 nM T94033 CJWE07 10368488 IC50 = 73 nM T94033 CDO83F 10368538 Ki = 210 nM T94033 C9ZD0S 10368685 Ki > 5000 nM T94033 CE27CV 10370457 Ki = 3 nM T94033 CHM7I1 10385552 IC50 = 5100 nM T94033 CYBF76 10386378 Ki > 50000 nM T94033 C26CSM 10386393 IC50 = 18 nM T94033 C71PIO 10387118 Ki = 7.8 nM T94033 C7TH5Q 10387956 Ki = 1200 nM T94033 CMNP39 10389039 IC50 > 10000 nM T94033 CLGF71 10389462 Ki = 4240 nM T94033 CE45NM 10389524 Ki = 900 nM T94033 CL3F1U 10389579 Ki = 3300 nM T94033 CM6L0W 10389769 Ki = 68500 nM T94033 C47OZV 10390121 Ki = 0.06 nM T94033 CSC52L 10390341 Ki = 6.2 nM T94033 C8EPN7 10390481 Ki = 8 nM T94033 C3BR5A 10390490 Ki = 0.25 nM T94033 CXF20B 10391310 IC50 = 15 nM T94033 CJNV62 10391699 IC50 > 33000 nM T94033 C6S4CO 10391715 Ki = 960 nM T94033 CEH4D1 10391881 IC50 = 230 nM T94033 CLK08Z 10391999 IC50 > 10000 nM T94033 C7QYK4 10392081 IC50 > 300000 nM T94033 CF6P1M 10392348 Ki = 4300 nM T94033 CNMD35 10393290 Ki = 1400 nM T94033 C9BW6F 10393336 Ki = 0.86 nM T94033 CPQY05 10393804 Ki = 93 nM T94033 CCA45U 10394183 IC50 = 510 nM T94033 CM1WJ6 10394292 Ki = 2600 nM T94033 C6TS5H 10408877 IC50 = 250 nM T94033 C4FBO0 10409093 Ki = 3.3 nM T94033 C56NXW 10409551 IC50 = 3100 nM T94033 CC67OS 10409569 Ki = 150 nM T94033 CO3Z5D 10409945 IC50 = 36000 nM T94033 CMQY61 10410471 Ki = 130 nM T94033 C2L8SQ 10410499 IC50 = 38000 nM T94033 C9AM3R 10410743 IC50 > 10000 nM T94033 CL34IB 10410866 Ki = 1000 nM T94033 C70AME 10411443 IC50 > 10000 nM T94033 C20ZSL 10411684 Ki > 5000 nM T94033 CYZ4O1 10411843 IC50 = 11 nM T94033 CD0VI1 10412365 IC50 = 370 nM T94033 CE61DA 10413099 IC50 = 1.5 nM T94033 C03MWI 10413130 Ki = 1180 nM T94033 CXU03I 10413657 Ki = 530 nM T94033 CW73XP 10414157 Ki = 0.9 nM T94033 CVG67Q 10414711 Ki = 130 nM T94033 CT57QN 10414868 IC50 = 23 nM T94033 CF8M6C 10415115 Ki = 2900 nM T94033 C2E3XM 10417117 Ki = 1.2 nM T94033 CB4X5P 10417378 Ki = 42200 nM T94033 CVK4L6 10418061 IC50 = 1600 nM T94033 CBV6N7 10423722 IC50 > 50000 nM T94033 CJTH60 10432907 Ki = 21600 nM T94033 C1RE8V 10433463 IC50 > 10000 nM T94033 C4K9QX 10433872 IC50 > 10000 nM T94033 CK3YW7 10434792 Ki = 60 nM T94033 CX39AB 10435238 Ki = 3100 nM T94033 CHCI84 10435532 Ki = 380 nM T94033 C48HDV 10435701 Ki = 0.4 nM T94033 CLSC78 10436040 Ki = 2.6 nM T94033 C9K5GO 10436126 Ki = 0.05 nM T94033 CUM2T7 10436294 Ki = 7400 nM T94033 CG07WY 10438196 Ki = 300 nM T94033 C1YA8S 10438982 Ki = 110 nM T94033 C4XD5V 10439687 Ki = 102000 nM T94033 C0AU7M 10441103 IC50 = 8700 nM T94033 CL4K2S 10447733 IC50 > 200000 nM T94033 CXYZ72 10453194 Ki = 1.5 nM T94033 CCU35L 10453208 IC50 > 10000 nM T94033 C8D3IZ 10453647 Ki = 670 nM T94033 C9M5RI 10453763 Ki = 230 nM T94033 C4SZV0 10454685 Ki = 15900 nM T94033 C7HOX3 10454867 IC50 = 21000 nM T94033 CV9N1X 10457101 Ki = 1.5 nM T94033 CS1O2X 10458005 Ki = 3.3 nM T94033 C50FMX 10458597 Ki = 170 nM T94033 C43UIL 10459664 Ki = 19 nM T94033 COU03P 10459896 IC50 = 18 nM T94033 C9W5IS 10460210 Ki = 7400 nM T94033 C9HI6A 10460541 IC50 = 829 nM T94033 CI87FD 10460564 IC50 > 2500 nM T94033 C6KJM2 10461790 Ki > 50000 nM T94033 CJW85F 10461946 Ki = 22 nM T94033 CQ4AF3 10462372 IC50 = 1900 nM T94033 CWG91R 10472893 Ki > 25000 nM T94033 CO8A1D 10475379 Ki = 9 nM T94033 CKJ46M 10476712 Ki = 69 nM T94033 C7O6BE 10477973 Ki = 16 nM T94033 C0W7NM 10478661 Ki = 220 nM T94033 CZO69X 10478912 IC50 = 40 nM T94033 C63GRO 10479438 IC50 = 0.98 nM T94033 C6T3LA 10479448 Ki = 0.4 nM T94033 C2BOG5 10479744 IC50 = 8 nM T94033 C1MX6F 10480245 Ki = 200 nM T94033 C45KWI 10480373 Ki = 500 nM T94033 CCP2N8 10480374 Ki > 4000 nM T94033 CV0X6G 10480463 IC50 > 11000 nM T94033 CF2G8Q 10481025 Ki = 1200 nM T94033 CM5A3J 10481558 Ki = 3000 nM T94033 CMIN26 10481978 Ki = 200 nM T94033 CRY09K 10482192 IC50 = 1700 nM T94033 CI45GW 10482478 Ki = 0.9 nM T94033 C9F8PU 10482918 Ki = 3.2 nM T94033 CG18KR 10483116 Ki = 13 nM T94033 CJ50AY 10483408 Ki = 500 nM T94033 C3SGO9 10483470 Ki = 86 nM T94033 CEI65Z 10483775 Ki = 12600 nM T94033 C7BN0W 10496623 IC50 = 1390 nM T94033 CKL8H3 10497634 Ki = 19200 nM T94033 CY8P5O 10500432 IC50 = 230 nM T94033 CQE12B 10501172 Ki = 120 nM T94033 C1F7IZ 10501283 Ki = 21500 nM T94033 C6F2ZX 10501400 Ki > 5000 nM T94033 CFU1E5 10501943 Ki = 740 nM T94033 CFP53Y 10502109 IC50 > 33000 nM T94033 CKI70V 10502393 Ki = 360 nM T94033 C2C4XR 10502821 IC50 = 106 nM T94033 CEKX36 10503075 Ki > 4000 nM T94033 C4O9JK 10503954 Ki > 4000 nM T94033 CY16UR 10504366 Ki = 1750 nM T94033 CXGK70 10505240 Ki = 20 nM T94033 CG5IS0 10505288 Ki = 210 nM T94033 C09TUO 10506433 Ki = 1080 nM T94033 CXL48O 10507039 Ki = 43 nM T94033 C7SU8I 10507339 Ki = 17 nM T94033 CXB50R 10508061 Ki = 1200 nM T94033 C5F8HM 10509332 IC50 = 13300 nM T94033 CT41HV 10509499 IC50 < 50000 nM T94033 CZ01JY 10511253 Ki = 1200 nM T94033 CF58EC 10515237 Ki = 348 nM T94033 C3XC0G 10517758 Ki = 120 nM T94033 C9S6NI 10522214 Ki = 565 nM T94033 CQS6Y2 10523322 Ki = 130 nM T94033 CKQ17F 10523978 IC50 = 9330 nM T94033 CFL49H 10524222 Ki = 2100 nM T94033 C87BCM 10525391 Ki = 1900 nM T94033 CJ15UC 10525392 Ki > 21000 nM T94033 CD82SZ 10525943 Ki > 5000 nM T94033 CZ0E8S 10526100 Ki = 11000 nM T94033 CE25ZS 10526243 IC50 > 132000 nM T94033 C42XPE 10526785 Ki = 2800 nM T94033 C7Y0WM 10527751 Ki > 4000 nM T94033 CS7UC4 10528210 Ki = 1900 nM T94033 CU8I0J 10528552 Ki = 800 nM T94033 CT41XW 10528653 Ki > 4000 nM T94033 C5ED3G 10529121 Ki = 0.61 nM T94033 CA0QG6 10531178 Ki = 900 nM T94033 C1K0NS 10532026 Ki = 2100 nM T94033 CKYZ01 10532259 Ki = 600 nM T94033 C43TPO 10536580 Ki = 107 nM T94033 C6TJ7O 10539116 Ki = 197 nM T94033 C0K6LY 10541776 Ki = 177 nM T94033 COB07E 10543987 Ki = 6200 nM T94033 CV1EL2 10544014 Ki = 210 nM T94033 CK13IY 10546004 Ki = 6500 nM T94033 CO1JW8 10546322 Ki = 120 nM T94033 CEP1L6 10547293 Ki = 1000 nM T94033 CO46GQ 10548215 Ki = 12850 nM T94033 CYEN07 10548429 Ki > 5000 nM T94033 C37BYS 10548542 Ki = 8.3 nM T94033 CEC7J6 10549325 Ki > 21000 nM T94033 C2F6CT 10549508 Ki = 1900 nM T94033 C4HF7I 10550428 IC50 = 60 nM T94033 CWLZ02 10550997 IC50 = 90 nM T94033 CB81VQ 10551446 Ki > 4000 nM T94033 CVR3P1 10552445 Ki = 4000 nM T94033 C4Q5VT 10552446 Ki = 180 nM T94033 CCM1I8 10552861 Ki = 16 nM T94033 C0ULI2 10553110 Ki = 18 nM T94033 CYX1V7 10553919 Ki = 954 nM T94033 C4J1KI 10554052 Ki > 4000 nM T94033 CT4F2L 10554762 Ki = 3.4 nM T94033 CG94EU 10554804 Ki = 403 nM T94033 CE8V0B 10555065 Ki = 3500 nM T94033 CWR8G9 10555769 Ki > 4000 nM T94033 CGQ38W 10555959 Ki = 5800 nM T94033 CQG10I 10556031 Ki = 810 nM T94033 CSK8V5 10556085 Ki > 21000 nM T94033 CGHL47 10556206 Ki = 4500 nM T94033 C38UHV 10559603 Ki = 890 nM T94033 CLT21Y 10561384 Ki = 99 nM T94033 CQ07NP 10564031 Ki = 202 nM T94033 CY1JF2 10569959 Ki = 8000 nM T94033 CZ6HD9 10570938 Ki = 3433 nM T94033 C52FQT 10571832 Ki = 1535 nM T94033 C6KO1H 10572047 IC50 = 910 nM T94033 C1HA7S 10572228 Ki = 1600 nM T94033 C2VG9M 10572774 Ki = 600 nM T94033 CV71RX 10573919 Ki = 1400 nM T94033 CS8H3A 10574097 Ki > 5000 nM T94033 CSHM62 10575806 Ki = 1200 nM T94033 CY5O2K 10576002 Ki > 5000 nM T94033 CY1A0X 10576138 Ki > 4000 nM T94033 CT8P9K 10578388 Ki = 360 nM T94033 CA16OW 10579010 Ki = 44 nM T94033 C9MN1H 10579028 Ki = 21000 nM T94033 C6LO8Q 10580222 Ki = 3000 nM T94033 C1D8GI 10580396 Ki = 500 nM T94033 C42LVU 10580437 Ki = 2000 nM T94033 CX1T3J 10586377 Ki = 103 nM T94033 C0SWO6 10586704 Ki = 132 nM T94033 C1XUT8 10589842 Ki = 154 nM T94033 C02RYN 10592155 Ki = 7700 nM T94033 C9GEN0 10593215 Ki = 243 nM T94033 CLP7V3 10593216 Ki = 177 nM T94033 CB5FH2 10593304 Ki = 520 nM T94033 C43PRO 10593976 IC50 > 300000 nM T94033 CTV74P 10594741 Ki = 169 nM T94033 C4VMO3 10595198 Ki = 3600 nM T94033 CWJ68A 10596601 Ki > 100000 nM T94033 CO3N1I 10597592 Ki > 4000 nM T94033 CI5CH1 10597827 Ki = 450 nM T94033 CT2E6F 10598802 Ki = 380 nM T94033 C8P3QI 10599262 Ki = 7 nM T94033 CJZF07 10599669 Ki > 4000 nM T94033 C3HI1S 10599710 Ki = 60 nM T94033 C7SEQ9 10599734 Ki > 4000 nM T94033 CD6L3E 10600145 Ki > 4000 nM T94033 CCQU28 10600245 Ki = 2100 nM T94033 C8L9FV 10600329 Ki > 4000 nM T94033 CVEH84 10600484 Ki = 10 nM T94033 C21PEX 10602709 Ki = 2400 nM T94033 CM4WU9 10602877 IC50 = 90 nM T94033 C76MXV 10602962 Ki = 0.1 nM T94033 CD8LW5 10603201 Ki = 60 nM T94033 C0SD6T 10603555 Ki = 12000 nM T94033 CW5BQ4 10603912 Ki = 15 nM T94033 CP69LR 10604270 Ki = 3100 nM T94033 C8CQY2 10604382 Ki = 50 nM T94033 CY1J0N 10604774 Ki = 70 nM T94033 CY91TB 10609450 Ki = 88 nM T94033 C8ZXS3 10609754 IC50 = 10 nM T94033 CV12FZ 10611202 Ki = 112 nM T94033 CLD32T 10611279 Ki = 96 nM T94033 CV4RZ9 10611280 Ki = 219 nM T94033 CAWH91 10611651 Ki = 147 nM T94033 CAM89Z 10614687 Ki = 138 nM T94033 C1RH3P 10621200 Ki = 3100 nM T94033 CC26YF 10622456 Ki > 5000 nM T94033 CO83BP 10622800 IC50 = 1200 nM T94033 C39IFP 10623057 Ki > 4000 nM T94033 C5K8QJ 10623402 Ki = 350 nM T94033 CXD95O 10623670 Ki > 5000 nM T94033 CSP20T 10623756 Ki = 2400 nM T94033 CZJL67 10623842 Ki = 2228 nM T94033 CV0I5Y 10623890 Ki = 14000 nM T94033 C3OJ4U 10623965 Ki = 300 nM T94033 C69VAT 10624206 Ki = 2600 nM T94033 C1ZW5F 10624489 Ki = 2500 nM T94033 CH3A1M 10625087 Ki = 50 nM T94033 CB2X5R 10625525 Ki = 50 nM T94033 C8S6QZ 10625945 Ki > 4000 nM T94033 C8PHU2 10626697 Ki = 560 nM T94033 CJ62ZG 10626722 Ki = 350 nM T94033 CK25AY 10626893 Ki = 3.6 nM T94033 C8K7RA 10627065 Ki = 27 nM T94033 CMP4X2 10627067 Ki = 15 nM T94033 CQ7F0T 10627268 Ki = 14000 nM T94033 C03CIN 10628066 Ki = 10000 nM T94033 C1BM4L 10636757 Ki = 152 nM T94033 C1PX0H 10642149 Ki = 810 nM T94033 CF3P4J 10642387 Ki > 5000 nM T94033 C8C5WU 10644578 IC50 = 13200 nM T94033 C4KMJ8 10644692 Ki = 3700 nM T94033 CZ9L8T 10644693 Ki = 1400 nM T94033 C4M0QB 10645022 Ki = 2000 nM T94033 C0QP4O 10645136 Ki > 4000 nM T94033 C3S0GW 10645345 Ki = 22000 nM T94033 CFNH06 10645807 IC50 = 3400 nM T94033 C72XTB 10646342 Ki = 630 nM T94033 CNC25X 10646757 Ki > 5000 nM T94033 CRMG36 10647285 Ki = 900 nM T94033 C1XDA6 10647609 IC50 = 31000 nM T94033 CR1Y2D 10647704 Ki = 1000 nM T94033 C76RFN 10647907 Ki = 1051 nM T94033 C1BG8S 10648377 Ki = 0.45 nM T94033 C41KHW 10648454 Ki = 201 nM T94033 C8N7VE 10650243 Ki = 8.1 nM T94033 C1KVB3 10650805 Ki = 510 nM T94033 C2OSA9 10651120 Ki = 130 nM T94033 C6E4WZ 10651873 Ki = 2800 nM T94033 CD2X1K 10652683 IC50 < 50000 nM T94033 CBHW74 10653967 Ki = 240 nM T94033 CMXS14 10653995 Ki > 15000 nM T94033 C4R6AH 10655867 Ki = 895 nM T94033 C13MSZ 10656555 Ki = 213 nM T94033 C8XK7P 10656953 Ki = 270 nM T94033 C42PDV 10658840 Ki = 325 nM T94033 CG40SW 10661464 Ki = 4400 nM T94033 C54ZOF 10661847 Ki = 170 nM T94033 CW75PO 10661946 IC50 > 100000 nM T94033 CBT96N 10664145 Ki > 10000000 nM T94033 CRDG85 10665326 Ki = 1200 nM T94033 CJH38X 10665512 IC50 = 870 nM T94033 CV5A3R 10667379 IC50 = 44700 nM T94033 C4WCH6 10668443 Ki > 5000 nM T94033 CJG9H6 10669349 Ki = 5 nM T94033 CUD8A7 10669525 Ki = 2500 nM T94033 C7CVW2 10669933 IC50 = 2200 nM T94033 C9MUX3 10670446 IC50 = 57 nM T94033 CD2C0U 10670479 Ki = 1700 nM T94033 C6PAD8 10670666 Ki > 4000 nM T94033 CZO1K8 10671210 Ki = 1960 nM T94033 C3FHO0 10671226 Ki = 2.5 nM T94033 C4LJO3 10671702 Ki = 70 nM T94033 CIKJ09 10672223 Ki = 1700 nM T94033 CW1G9B 10672666 IC50 > 10000 nM T94033 C56NHZ 10674014 IC50 = 18 nM T94033 CM1Y2D 10675086 Ki = 2800 nM T94033 C82NMW 10675362 Ki = 21 nM T94033 C4TIU1 10675632 Ki = 70 nM T94033 C8P2UC 10675884 Ki = 3100 nM T94033 CXL4W8 10679763 Ki = 185 nM T94033 CO37WG 10680915 Ki = 106 nM T94033 CO46RX 10682070 Ki = 136 nM T94033 CZM7X9 10682615 Ki = 205 nM T94033 CD3H4Q 10682687 Ki = 355 nM T94033 CQWI96 10683513 Ki = 172 nM T94033 CFQ5V2 10690751 Ki = 350 nM T94033 C3KL1Y 10691215 IC50 = 140 nM T94033 CVE95Z 10691360 Ki = 37000 nM T94033 CI48CW 10692578 Ki > 5000 nM T94033 CD8S2B 10692579 Ki = 4200 nM T94033 C7IU6Y 10692676 Ki = 2.5 nM T94033 CID1F6 10693808 Ki = 5100 nM T94033 CZ53XC 10693841 Ki > 5000 nM T94033 CS08UM 10694720 Ki > 5000 nM T94033 CVR1F9 10694772 Ki > 4000 nM T94033 CJPN01 10694782 Ki = 0.1 nM T94033 CIB63V 10694800 Ki = 6800 nM T94033 CC35DA 10695507 IC50 > 33000 nM T94033 CW8RV0 10696389 Ki = 400 nM T94033 CP4QC5 10696511 Ki = 3 nM T94033 CKD68U 10696697 Ki = 2.1 nM T94033 C3QH0L 10697320 Ki = 4400 nM T94033 C3WC0Q 10698376 Ki = 380 nM T94033 CWX87E 10698758 Ki = 360 nM T94033 C8IUF9 10699264 Ki = 19 nM T94033 C9DRY5 10705378 Ki = 121 nM T94033 C4CNK6 10706336 Ki = 97 nM T94033 CY0P5F 10714145 Ki = 4700 nM T94033 CF6TZ2 10715258 Ki = 2800 nM T94033 CK2WI6 10715476 Ki = 27000 nM T94033 CZB24K 10715861 Ki > 5000 nM T94033 C0TE1Z 10716448 Ki = 12600 nM T94033 C49JDV 10717698 Ki = 630 nM T94033 CFG6T3 10717789 Ki = 1340 nM T94033 CCP58N 10718840 Ki = 900 nM T94033 C82FPL 10718889 Ki > 4000 nM T94033 CFH75T 10718950 Ki > 4000 nM T94033 C1Z3PF 10719336 Ki = 1400 nM T94033 COA5Z1 10719523 Ki = 880 nM T94033 CIKF89 10719580 Ki = 14 nM T94033 CJ8TN7 10720504 Ki = 6 nM T94033 CLXN90 10721219 Ki = 440 nM T94033 C9O7LM 10721366 Ki = 17 nM T94033 C0OER6 10721605 Ki = 3000 nM T94033 CMUX37 10722043 Ki = 2100 nM T94033 C69IHQ 10722538 Ki = 15 nM T94033 CAS17I 10722747 Ki = 5000 nM T94033 CUTA38 10723163 Ki = 100 nM T94033 CR06TK 10724264 IC50 = 18200 nM T94033 CV3W6Y 10732869 Ki = 98 nM T94033 CL29UP 10737764 IC50 = 1510 nM T94033 CF9VZ0 10738109 Ki > 500 nM T94033 CZ0G6W 10738922 Ki = 200 nM T94033 C1GCY4 10739768 Ki = 290 nM T94033 CL7RC5 10742017 IC50 > 33000 nM T94033 C64AUD 10742143 Ki = 4000 nM T94033 CZ0Q8K 10742217 Ki = 0.5 nM T94033 CK26FW 10742542 Ki = 1300 nM T94033 CQ26JG 10744246 Ki = 30 nM T94033 CO3NI6 10744295 Ki = 62 nM T94033 C7RWD8 10744643 Ki = 0.31 nM T94033 C5L7HE 10745242 Ki = 900 nM T94033 CAUM51 10745299 Ki = 200 nM T94033 CU5OG9 10746409 Ki = 751 nM T94033 C3V8JP 10746573 Ki = 300 nM T94033 C93QXR 10747940 IC50 = 17800 nM T94033 CK4PG1 10752795 Ki = 276 nM T94033 CWLF28 10753747 Ki = 166 nM T94033 C8J9PM 10761427 Ki = 1200 nM T94033 C9JLQ7 10761484 Ki = 19600 nM T94033 CHA46Q 10764382 Ki = 600 nM T94033 C0FTS9 10764466 Ki > 5000 nM T94033 C9SDJ1 10765420 Ki = 2600 nM T94033 CD51XL 10765919 Ki > 4000 nM T94033 CQUM96 10765972 Ki = 1600 nM T94033 CQ5F1A 10767215 Ki = 39 nM T94033 CJSW62 10767268 Ki > 4000 nM T94033 C9SQB5 10767957 Ki = 300 nM T94033 CZWC95 10768463 Ki = 2000 nM T94033 C6CT4O 10768464 Ki = 0.4 nM T94033 CCK3E5 10768801 Ki = 263 nM T94033 C5DYQ3 10769476 Ki = 6000 nM T94033 C62KFB 10769759 Ki = 8100 nM T94033 C24ZSE 10769921 Ki > 2000 nM T94033 C5E6AY 10770527 Ki = 4300 nM T94033 C4Z2LQ 10770606 Ki = 3400 nM T94033 CQW74C 10770621 Ki = 2900 nM T94033 CCZ9U0 10770773 Ki = 300 nM T94033 C3W7TF 10770845 Ki = 5800 nM T94033 CBH54X 10771811 Ki = 5300 nM T94033 C7HJW8 10775754 Ki = 240 nM T94033 CEIV75 10779010 Ki = 160 nM T94033 C7VXA1 10784195 Ki = 8500 nM T94033 CJ04LS 10784328 IC50 = 6030 nM T94033 C2IBK7 10784421 IC50 = 230 nM T94033 CJ7O1H 10785523 Ki = 1400 nM T94033 C7BRQ1 10785917 IC50 > 132000 nM T94033 CI9BZ1 10786604 Ki = 6000 nM T94033 CQRZ02 10787180 Ki = 350 nM T94033 CD1CF3 10787181 Ki = 3700 nM T94033 C0AUV8 10788046 Ki = 4400 nM T94033 C4CAT2 10788047 Ki = 1100 nM T94033 CRHE34 10788206 Ki > 5000 nM T94033 CD21MW 10788364 Ki > 4000 nM T94033 C2KOA4 10788644 Ki = 10300 nM T94033 CKLU46 10788963 Ki = 325 nM T94033 CQU20Z 10789503 IC50 = 190 nM T94033 CJZ35V 10789732 Ki = 3 nM T94033 C0RL4C 10789777 Ki > 4000 nM T94033 CMX5V9 10789805 Ki > 4000 nM T94033 CT8M1C 10790019 Ki > 21000 nM T94033 CG73DE 10790153 Ki = 440 nM T94033 CL73OX 10791003 Ki = 3.9 nM T94033 CXYB12 10791358 Ki = 40 nM T94033 C5TID3 10791816 Ki > 4000 nM T94033 CBNP58 10792157 Ki = 1500 nM T94033 CRD65S 10792619 Ki = 7.6 nM T94033 C89CFX 10793224 Ki = 239 nM T94033 CLWY92 10793236 Ki = 110 nM T94033 CL7M3H 10793760 Ki = 18 nM T94033 C5ENU2 10794450 Ki = 900 nM T94033 C64ZVF 10794532 Ki = 3800 nM T94033 CC95IV 10794535 Ki = 1300 nM T94033 CR5A3Q 10799358 Ki = 450 nM T94033 C60CFR 10799567 Ki = 280 nM T94033 CS7PH9 10801237 Ki = 189 nM T94033 C5XAK8 10801238 Ki = 213 nM T94033 CU43PJ 10801239 Ki = 324 nM T94033 CN05LQ 10801551 Ki = 154 nM T94033 C8AP1D 10804436 Ki = 153 nM T94033 CD6U1P 10806942 Ki > 4200 nM T94033 C1HJ7R 10807538 Ki = 134 nM T94033 CYAJ14 10810195 Ki = 300 nM T94033 CL9O0C 10810196 Ki = 360 nM T94033 CUQX02 10810754 Ki = 630 nM T94033 C0U7PJ 10811747 Ki = 150 nM T94033 CI70OG 10811911 IC50 = 380 nM T94033 C81HPC 10812830 IC50 = 20400 nM T94033 CYS08X 10813043 Ki = 2300 nM T94033 CX6YF7 10813081 Ki = 19500 nM T94033 C4YA1H 10813083 Ki = 62400 nM T94033 CQK97I 10813230 Ki > 4000 nM T94033 C3WX4F 10813359 Ki = 2200 nM T94033 C13KAX 10813709 Ki = 1500 nM T94033 CZA0D1 10814968 Ki = 230 nM T94033 CE1DT2 10815540 Ki = 1440 nM T94033 CV1U5L 10816337 Ki = 1160 nM T94033 CL8YB0 10816451 Ki = 970 nM T94033 CC9LF3 10816800 Ki = 21 nM T94033 CPRS52 10817210 Ki = 3 nM T94033 CSZR21 10817699 Ki = 16000 nM T94033 CUS6D0 10818009 Ki = 10800 nM T94033 CB5E9C 10818749 IC50 = 130 nM T94033 C21RNT 10819005 IC50 = 70 nM T94033 CIR3E1 10819322 IC50 = 900 nM T94033 CG9B1J 10819798 Ki > 15000 nM T94033 C2D1KY 10820951 IC50 > 50 nM T94033 CZHW69 10821268 Ki = 1365 nM T94033 C0QR1N 10822474 Ki = 330 nM T94033 C6TU4I 10824479 Ki = 266 nM T94033 CD2C8Y 10825077 Ki = 133 nM T94033 CC8W0O 10827539 Ki = 265 nM T94033 C0M3XB 10831506 Ki = 14000 nM T94033 CE2LP4 10832026 Ki > 5000 nM T94033 CLXP56 10833102 Ki = 2100 nM T94033 CYAG10 10834106 IC50 = 120 nM T94033 CJ2M4I 10835535 Ki > 5000 nM T94033 CW8OT1 10835646 Ki > 5000 nM T94033 CJ0KB8 10835917 Ki = 22 nM T94033 C2KXJ7 10835995 Ki > 4000 nM T94033 CH0RG9 10836919 Ki > 4000 nM T94033 C67FIC 10837478 Ki = 3000 nM T94033 CW3YA2 10837929 Ki = 3400 nM T94033 C1FTR2 10837980 Ki = 278 nM T94033 C5FSB0 10838473 Ki = 3400 nM T94033 CCH6W7 10840002 Ki = 9.6 nM T94033 C7G3LP 10840570 Ki = 225 nM T94033 CM13CR 10840852 Ki = 200 nM T94033 CYX51H 10840933 Ki = 3900 nM T94033 CZVR32 10841125 Ki = 9 nM T94033 COLC79 10841532 Ki = 11 nM T94033 C6QF7T 10841535 Ki = 1450 nM T94033 C2R7OQ 10841758 Ki = 2100 nM T94033 C6DVC1 10846955 Ki = 328 nM T94033 CLMB72 10847696 Ki = 255 nM T94033 CB94KC 10847800 Ki = 104 nM T94033 CBK06L 10861643 IC50 > 100000 nM T94033 CWLR90 10862090 IC50 = 28000 nM T94033 CP5D7Z 10862803 Ki = 0.14 nM T94033 CB38YZ 10863406 Ki > 5000 nM T94033 CV8AO7 10863550 Ki = 3.5 nM T94033 CK7VC8 10863579 Ki > 5000 nM T94033 CZHE72 10863632 IC50 = 10000 nM T94033 CKG30N 10863633 Ki = 7.9 nM T94033 CN6WO8 10863757 Ki = 1.3 nM T94033 C80QUN 10863817 Ki = 90000 nM T94033 C07BLI 10864217 Ki = 2070 nM T94033 CL5C1N 10864452 Ki = 0.82 nM T94033 C2E8FZ 10864521 IC50 = 580 nM T94033 C62IPV 10864710 Ki = 540000 nM T94033 C02XLH 10865109 IC50 = 40 nM T94033 CZX59B 10865289 Ki = 28000 nM T94033 C9LEJ0 10865386 IC50 = 15400 nM T94033 C1BOZ5 10865461 IC50 = 14600 nM T94033 CN2CE8 10865462 IC50 = 3420 nM T94033 CLB15C 10871563 Ki > 75000 nM T94033 CF59UR 10873499 IC50 = 1600 nM T94033 CBP8H5 10873750 IC50 = 1300 nM T94033 CD7I4A 10873871 Ki > 5000 nM T94033 CI3C1A 10874054 IC50 = 210 nM T94033 C0KIZ5 10874086 Ki > 5000 nM T94033 C80TLH 10874136 IC50 = 10600 nM T94033 CQ5E9L 10874168 Ki = 146 nM T94033 CXG62W 10874449 Ki > 3900 nM T94033 C2TH3I 10875009 Ki > 3900 nM T94033 CXT8N6 10875598 IC50 = 4400 nM T94033 C7YEP4 10875960 IC50 = 100000 nM T94033 C80WCU 10883641 Ki > 5000 nM T94033 C7Z2BD 10883660 IC50 = 16000 nM T94033 CN74ZX 10884041 Ki = 0.54 nM T94033 C19DGJ 10884304 Ki = 1.1 nM T94033 CP4V1J 10885177 IC50 = 600 nM T94033 C1PNQ4 10885181 Ki > 5000 nM T94033 CKB5P1 10885309 Ki = 0.33 nM T94033 CCH3S0 10885334 IC50 > 30000 nM T94033 CVK67J 10885344 Ki = 0.29 nM T94033 C38EXQ 10885426 IC50 > 100000 nM T94033 C27LWG 10885612 Ki = 270 nM T94033 C2MV8C 10886082 IC50 = 14000 nM T94033 CU8J0C 10894269 Ki > 1500000 nM T94033 CJGS43 10894874 Ki = 38000 nM T94033 C49BRD 10894895 Ki = 950 nM T94033 C1VRY3 10895218 Ki = 4.8 nM T94033 CW1KL6 10895606 Ki > 1000 nM T94033 C1V2QA 10895649 IC50 = 73 nM T94033 CW7Q2U 10895700 IC50 > 2500 nM T94033 C3FD4T 10895707 IC50 = 20000 nM T94033 C3OJF7 10895978 IC50 = 1790 nM T94033 C16NXJ 10896126 Ki = 480 nM T94033 CMU96G 10896304 IC50 = 16500 nM T94033 CMP45U 10896308 Ki > 21000 nM T94033 CJ4D9G 10896528 IC50 > 100000 nM T94033 C1CYR0 10896771 Ki = 0.015 nM T94033 C39AVR 10897080 Ki = 9090 nM T94033 C3X1JV 10897344 IC50 = 100 nM T94033 C59ETF 10897550 Ki = 3900 nM T94033 C2GPU4 10897682 IC50 = 440 nM T94033 CQTC02 10903566 Ki = 7000 nM T94033 CUMI91 10905246 Ki = 280 nM T94033 CDWX72 10905375 IC50 = 58884.37 nM T94033 C9AD3P 10905499 IC50 = 3400 nM T94033 CB1HW4 10905809 IC50 > 30000 nM T94033 COX30Q 10905999 IC50 = 390 nM T94033 C3ZY5O 10906286 IC50 = 23000 nM T94033 C7E3AJ 10906300 Ki = 9.8 nM T94033 C9C6UE 10906426 Ki > 21000 nM T94033 CH2G5Q 10906977 Ki = 1900 nM T94033 CTM36K 10907121 Ki > 5000 nM T94033 CQ6OM5 10907189 IC50 = 2800 nM T94033 CZU8X9 10908149 IC50 = 36200 nM T94033 CPJ1Q7 10908669 IC50 = 12000 nM T94033 C9E7RY 10908791 IC50 = 4990 nM T94033 C2BXU9 10908808 IC50 = 4590 nM T94033 CC19NT 10915968 Ki = 1585 nM T94033 C5I7SU 10916321 Ki > 5000 nM T94033 CA1IB4 10916653 Ki > 5000 nM T94033 CR8N0G 10917057 IC50 = 2400 nM T94033 CW84NP 10917410 IC50 = 60 nM T94033 CY95IG 10917479 IC50 = 330 nM T94033 CG32HJ 10917579 Ki = 13 nM T94033 C7K5SQ 10918066 Ki > 5000 nM T94033 CT82AP 10918697 Ki = 0.02 nM T94033 C57GDA 10918949 IC50 = 8600 nM T94033 C7A5FP 10919302 Ki = 30700 nM T94033 C5A8NU 10919581 IC50 = 7480 nM T94033 CK68OT 10927655 Ki = 1.6 nM T94033 C2G5RX 10927936 IC50 = 24000 nM T94033 CKI49C 10928313 Ki > 21000 nM T94033 CR5VW1 10928435 Ki = 200 nM T94033 C3OV9B 10928554 IC50 = 54 nM T94033 C5KM8X 10928726 Ki = 0.96 nM T94033 CJR8U5 10929318 Ki = 376 nM T94033 C3XL4K 10929422 Ki = 2.6 nM T94033 C5ODK4 10929522 Ki = 0.6 nM T94033 C1KV7H 10929853 Ki = 11900 nM T94033 C1Q9WZ 10930326 IC50 = 9200 nM T94033 CL20KX 10930722 IC50 = 1680 nM T94033 CE6W2Q 10938705 IC50 = 250 nM T94033 C8RF5U 10938960 Ki = 5300 nM T94033 CDWG32 10938987 Ki = 1.1 nM T94033 CMD6C0 10939317 Ki = 8000 nM T94033 CC81OU 10939381 Ki > 5000 nM T94033 CLAR40 10939595 Ki = 0.5 nM T94033 CDSU98 10939678 Ki > 5000 nM T94033 CBN2H7 10939759 IC50 > 30000 nM T94033 CNF69S 10939771 IC50 = 4250 nM T94033 C38WQM 10939772 IC50 > 30000 nM T94033 CW2K4T 10940667 Ki = 0.12 nM T94033 C8OA1L 10946869 Ki = 32000 nM T94033 CUN98K 10949030 Ki = 1800 nM T94033 CCM7H1 10949960 Ki = 730 nM T94033 C95WOX 10950363 Ki = 3800 nM T94033 CWN81P 10950417 Ki = 290 nM T94033 C5LS9R 10950524 IC50 = 13600 nM T94033 C2R1TW 10950927 IC50 = 1800 nM T94033 CE5SG3 10951082 IC50 > 100000 nM T94033 CT3BN9 10951324 Ki = 680000 nM T94033 CL5RI9 10951551 IC50 = 4000 nM T94033 CT6Z1I 10951552 IC50 = 300 nM T94033 CW85JZ 10951681 IC50 > 30000 nM T94033 C2TBO9 10959252 Ki > 75000 nM T94033 C9LJ7X 10960901 Ki > 1000 nM T94033 CB9KP4 10961420 Ki = 140000 nM T94033 CU17MI 10961677 IC50 = 35600 nM T94033 CY93FP 10961694 IC50 = 510 nM T94033 C18XBU 10961900 IC50 = 10000 nM T94033 CB07KT 10962223 Ki = 0.42 nM T94033 CITU70 10962439 Ki = 380 nM T94033 CQ5NX9 10962508 IC50 = 1100 nM T94033 CPQ2O9 10962541 IC50 > 30000 nM T94033 C3M9LW 10962721 IC50 = 130 nM T94033 CCE31H 10963578 IC50 = 3150 nM T94033 CWQ91E 10972679 IC50 < 40 nM T94033 CT6Q7Z 10972928 Ki = 1710 nM T94033 CJG58A 10973478 IC50 = 100 nM T94033 C89OXD 10973578 IC50 = 32 nM T94033 CC32DG 10973648 IC50 = 200 nM T94033 CB1JL6 10973926 IC50 = 6300 nM T94033 C6HG4P 10974490 IC50 = 24200 nM T94033 CVT26S 10974535 IC50 = 10400 nM T94033 CH41ZW 10974733 IC50 = 9920 nM T94033 CS1AL4 10983261 Ki = 7.1 nM T94033 CQGL23 10983472 Ki = 15 nM T94033 C9WO8T 10983680 IC50 = 8000 nM T94033 CPQ6O8 10983726 IC50 = 10 nM T94033 CJLX34 10983850 IC50 > 30000 nM T94033 C5DZA3 10984047 IC50 = 2000 nM T94033 CL9V7T 10984300 Ki > 3900 nM T94033 CJFO68 10984364 Ki = 0.43 nM T94033 CWVR40 10985371 IC50 = 12900 nM T94033 CWB42X 10993508 IC50 = 7800 nM T94033 CDP6C9 10994256 IC50 = 54700 nM T94033 CVI57D 10994262 Ki = 1.1 nM T94033 C8L3IJ 10994665 IC50 = 11220.18 nM T94033 C2DOM5 10995059 Ki = 0.1 nM T94033 CVMC01 10995072 Ki = 0.64 nM T94033 CS8Z9Q 10995111 Ki = 270 nM T94033 CZM0S7 10995244 Ki = 0.005 nM T94033 C84YIE 10995256 Ki = 0.16 nM T94033 CT7L2Q 10996309 IC50 = 84900 nM T94033 CH4B9C 11003663 IC50 = 58000 nM T94033 CUV8Q3 11004075 Ki = 0.27 nM T94033 C43SNO 11004109 Ki = 320 nM T94033 CF26JG 11004176 Ki > 5000 nM T94033 CK3N5I 11004200 Ki = 5300 nM T94033 C7FP6L 11004280 Ki = 140 nM T94033 C0RT9G 11004671 IC50 = 220 nM T94033 CP68KV 11004693 Ki > 5000 nM T94033 C7JQ3S 11005330 Ki = 1.8 nM T94033 CT8JY3 11005359 IC50 = 933.25 nM T94033 C5Y4LN 11005385 IC50 = 45400 nM T94033 CWHG91 11005419 Ki > 5000 nM T94033 CJF64C 11005941 IC50 = 900 nM T94033 CV3S4I 11006026 IC50 > 30000 nM T94033 CU4W0Z 11006040 Ki = 0.02 nM T94033 C9IBY6 11006214 IC50 = 1100 nM T94033 C9FU2Y 11006311 IC50 = 110 nM T94033 CC39SB 11009950 Ki = 340000 nM T94033 C3HW2I 11014107 Ki > 5000 nM T94033 CYZL25 11015002 Ki = 1400 nM T94033 C79NFR 11015314 IC50 = 120 nM T94033 CL5OG7 11015691 IC50 = 34400 nM T94033 C56HDX 11015700 Ki > 5000 nM T94033 C8I1VX 11016071 IC50 = 4600 nM T94033 CKW1O0 11016112 IC50 = 6980 nM T94033 CG71MR 11016812 IC50 = 37000 nM T94033 C69FOW 11025238 Ki = 1200 nM T94033 C4IE3S 11026399 Ki = 6.8 nM T94033 CYKF85 11026584 Ki > 5000 nM T94033 C21MKH 11026850 Ki > 5000 nM T94033 C46ZEX 11027375 Ki > 21000 nM T94033 C2RG6V 11028969 IC50 = 6820 nM T94033 CWJM96 11035993 IC50 = 19000 nM T94033 C3QG7H 11036285 Ki = 110000 nM T94033 CV1F8Q 11036379 Ki > 1500000 nM T94033 C80WPR 11036969 IC50 = 630 nM T94033 C5KTL2 11037540 Ki = 5600 nM T94033 C76BQW 11037740 IC50 = 8700 nM T94033 CIS2G7 11037772 IC50 = 5200 nM T94033 C4ZPT7 11037871 Ki = 370 nM T94033 CDI59J 11039222 IC50 > 30000 nM T94033 C7RM5W 11039881 IC50 = 11200 nM T94033 C7P5EN 11039916 IC50 > 30000 nM T94033 C9GPL1 11047203 IC50 > 130000 nM T94033 CMBL62 11048452 Ki = 3600 nM T94033 CYNU74 11048541 Ki = 1.2 nM T94033 CJL15S 11048586 Ki > 21000 nM T94033 CPEK84 11048789 Ki = 0.37 nM T94033 CF01BA 11049038 Ki > 21000 nM T94033 C4SW1T 11049045 Ki > 3900 nM T94033 CG2DO3 11049137 IC50 = 18700 nM T94033 CMV9L3 11049487 Ki = 0.21 nM T94033 COH39D 11049707 IC50 = 10000 nM T94033 C4UY7P 11050903 IC50 = 2400 nM T94033 CD9WJ8 11057540 Ki = 290 nM T94033 C2Y6VW 11057779 Ki = 110 nM T94033 C2RCQ3 11058560 IC50 = 680 nM T94033 CJZ10A 11059370 Ki > 21000 nM T94033 C7IA8Y 11059381 Ki = 4900 nM T94033 CZ43QG 11059512 Ki = 3000 nM T94033 CX09AC 11059549 Ki > 5000 nM T94033 CH1OX5 11059588 Ki = 2900 nM T94033 C8BC4U 11059598 Ki > 3900 nM T94033 CIT9A3 11059679 IC50 = 1230.27 nM T94033 CZ5OS9 11059701 IC50 = 27900 nM T94033 CXW4P2 11059783 Ki > 5000 nM T94033 CYG09F 11059945 Ki > 21000 nM T94033 CL01HN 11060467 IC50 = 23600 nM T94033 CRK76W 11060981 Ki = 15800 nM T94033 C3HNB2 11068806 Ki = 240 nM T94033 CVC69A 11069500 IC50 = 19000 nM T94033 CJ4U7M 11069959 Ki > 5000 nM T94033 C3HM5X 11070410 IC50 > 30000 nM T94033 CXC2Y3 11070493 IC50 = 10 nM T94033 C8ELX0 11070538 Ki = 120 nM T94033 C6R9ZK 11070689 IC50 = 10000 nM T94033 CP4R1J 11070822 Ki = 0.8 nM T94033 C30JDY 11071275 IC50 = 10000 nM T94033 C2IZ6R 11071363 IC50 = 8000 nM T94033 C5P4TB 11071386 Ki = 200 nM T94033 C5BS6T 11071397 Ki > 1000 nM T94033 CGM4D7 11071571 IC50 > 30000 nM T94033 CRQC89 11071685 IC50 = 15000 nM T94033 CK5PQ1 11072236 IC50 = 2000 nM T94033 C7YDH0 11072681 IC50 = 15400 nM T94033 CBW78D 11079334 IC50 = 130000 nM T94033 C29EIG 11079364 Ki = 17000 nM T94033 COU67Z 11079631 IC50 = 22000 nM T94033 CDKX73 11080299 Ki > 5000 nM T94033 CW3QV0 11080411 Ki > 5000 nM T94033 CM1XK2 11080560 IC50 = 1300 nM T94033 C4ISQ2 11080573 IC50 = 120000 nM T94033 CMJ61O 11080884 IC50 = 80600 nM T94033 CU63BK 11080954 IC50 = 3162.28 nM T94033 CSE89U 11081058 Ki > 3900 nM T94033 CZ73WT 11081112 Ki = 24000 nM T94033 C36HOU 11081121 IC50 = 19900 nM T94033 CCX29B 11081135 IC50 = 13000 nM T94033 CZLN21 11081488 IC50 > 100000 nM T94033 CNI4Y1 11081543 IC50 = 1200 nM T94033 CJ10SD 11082267 IC50 = 980 nM T94033 CVXQ65 11090840 IC50 = 93000 nM T94033 C2DFY6 11091090 IC50 = 940 nM T94033 CV0AS6 11091843 Ki = 3.6 nM T94033 C8QPS5 11092075 IC50 = 56234.13 nM T94033 CAW0O5 11092493 IC50 = 160 nM T94033 CJ6C3D 11092548 IC50 = 36800 nM T94033 CI74NM 11092809 IC50 = 4060 nM T94033 CULV92 11093279 Ki = 970 nM T94033 CACJ28 11101217 IC50 = 109000 nM T94033 CUTF06 11101863 IC50 = 2100 nM T94033 C9CUO6 11102065 IC50 = 7900 nM T94033 CIN7O0 11102236 IC50 > 30000 nM T94033 C2XAM1 11102245 Ki > 5000 nM T94033 CM1F6C 11102508 Ki > 5000 nM T94033 CVB8L0 11102692 Ki > 21000 nM T94033 C1GY8M 11102714 Ki > 5000 nM T94033 CQK68U 11103558 IC50 = 3300 nM T94033 CU53EA 11104490 IC50 = 15000 nM T94033 C41PZK 11112423 Ki = 300 nM T94033 C0L5YR 11112552 IC50 = 4600 nM T94033 C8JX1I 11113432 IC50 = 24000 nM T94033 CKL74M 11113517 Ki > 3900 nM T94033 C3Z0FD 11113624 IC50 = 3100 nM T94033 C30NPX 11113694 Ki > 21000 nM T94033 C0J4QW 11113965 IC50 > 200000 nM T94033 CI9VA0 11114013 Ki = 1.4 nM T94033 COT78V 11114139 IC50 = 300 nM T94033 C70RJC 11114562 IC50 = 3500 nM T94033 C7HI1X 11114579 Ki = 0.84 nM T94033 C4KRF5 11122174 IC50 = 38000 nM T94033 CEP79U 11122516 Ki > 5000 nM T94033 CDIS79 11122714 Ki > 5000 nM T94033 C03CFY 11122823 Ki = 2200 nM T94033 C4K6YA 11123202 Ki = 5.3 nM T94033 C0MKF7 11123270 IC50 = 4000 nM T94033 CJ54GQ 11123677 IC50 = 1000 nM T94033 C39ATZ 11124077 Ki > 21000 nM T94033 C72SVO 11124327 IC50 = 1200 nM T94033 C47UEP 11125405 IC50 = 50000 nM T94033 CD71SV 11125697 IC50 = 6300 nM T94033 CZYO41 11132865 IC50 > 130000 nM T94033 CMUG29 11133526 Ki = 1.4 nM T94033 CIH92Q 11133833 Ki > 1000 nM T94033 CT7S6O 11134002 Ki = 740 nM T94033 C8I6FL 11135396 IC50 = 720 nM T94033 CHI72V 11143925 IC50 = 3800 nM T94033 C8PK1N 11143992 IC50 = 350 nM T94033 C9KL8Y 11144992 Ki > 3900 nM T94033 CW84UN 11145308 IC50 = 17850 nM T94033 C8IU2S 11145990 IC50 = 7100 nM T94033 CDT6R4 11146027 Ki = 0.01 nM T94033 CIO01W 11146092 Ki = 2 nM T94033 C5MX1U 11146191 IC50 = 18900 nM T94033 CMX1S2 11146905 IC50 = 21700 nM T94033 CWMD96 11146965 IC50 = 28100 nM T94033 C1NMK4 11146971 IC50 = 9890 nM T94033 CAD15G 11149953 Ki = 17600 nM T94033 C96KWO 11155871 Ki = 19 nM T94033 CS1K9H 11156015 Ki = 71 nM T94033 CDPO91 11157107 Ki < 0.01 nM T94033 CQJG05 11157398 Ki = 4.5 nM T94033 C3W5PS 11157604 Ki = 1.6 nM T94033 CJ4X7R 11158066 IC50 = 500 nM T94033 C83DUK 11164311 IC50 > 10000 nM T94033 C5KG1A 11164549 Ki = 18200 nM T94033 C3WKQ1 11168297 Ki > 21000 nM T94033 CRG25K 11168660 IC50 > 10000 nM T94033 CV12FH 11168914 Ki = 0.018 nM T94033 CJ2X6P 11169058 Ki = 0.15 nM T94033 CZC46I 11179149 IC50 > 10000 nM T94033 CTM80Q 11179758 IC50 > 10000 nM T94033 CB23SU 11179962 Ki = 38 nM T94033 CU9K4E 11180045 IC50 = 560000 nM T94033 CEK78H 11181141 Ki = 0.042 nM T94033 C94SML 11181148 Ki = 53 nM T94033 C9X4JY 11181893 Ki = 600 nM T94033 C6LVG4 11186243 Ki = 35100 nM T94033 CTX9F3 11188793 Ki = 7310 nM T94033 CR0S7Z 11188883 Ki > 50000 nM T94033 C4V8ZF 11189887 Ki = 11 nM T94033 CU1BJ9 11191093 Ki = 0.25 nM T94033 CY70EN 11191165 IC50 > 10000 nM T94033 C7JS3U 11192255 Ki = 920 nM T94033 C5DSG6 11192607 Ki = 0.2 nM T94033 CZY84E 11192609 Ki = 0.3 nM T94033 CWA6L1 11202766 IC50 > 10000 nM T94033 CAM0I3 11203305 Ki > 25000 nM T94033 C93KMI 11203798 Ki = 1450 nM T94033 CJ6CW4 11203935 Ki > 21000 nM T94033 CA70NV 11214844 Ki = 7100 nM T94033 CKH8E1 11215005 Ki > 25000 nM T94033 CK3B9O 11215345 Ki = 0.14 nM T94033 C2K6HI 11215381 Ki = 15 nM T94033 CCS68P 11225163 Ki = 1.7 nM T94033 C8BRJ1 11225386 Ki > 21000 nM T94033 CK91AY 11225498 Ki = 0.66 nM T94033 CYV4U3 11225789 Ki = 5.6 nM T94033 C7DJT1 11226460 Ki > 25000 nM T94033 CP51FI 11226542 Ki = 9100 nM T94033 CSH3Y8 11226592 Ki = 110 nM T94033 CARW58 11227031 IC50 1 nM T94033 CJ4X0D 11236372 Ki = 0.77 nM T94033 CVK0I4 11237021 IC50 > 10000 nM T94033 CLA93S 11237163 Ki > 12000 nM T94033 C19KOM 11238809 IC50 = 0.3 ug.mL-1 T94033 CHLK70 11244460 Ki = 2350 nM T94033 C98HOZ 11249318 Ki = 4100 nM T94033 C5NZC6 11250356 Ki = 1.1 nM T94033 CL4JX3 11259447 Ki = 0.79 nM T94033 CHQ50D 11260319 IC50 > 10000 nM T94033 C7WIZ3 11261098 IC50 > 10000 nM T94033 CS2P9N 11261159 Ki = 3500 nM T94033 C2AFH8 11271916 IC50 > 10000 nM T94033 CRDU42 11271947 Ki > 25000 nM T94033 CA32ZV 11272101 IC50 = 915 nM T94033 CYRO76 11272254 IC50 = 2900 nM T94033 CW4OK6 11272980 Ki > 25000 nM T94033 CQFP08 11273559 Ki = 550 nM T94033 C73WSC 11273795 IC50 = 876 nM T94033 CB5RC4 11274304 Ki = 170 nM T94033 CON0H5 11283664 Ki = 0.65 nM T94033 CSH76U 11284767 Ki = 3700 nM T94033 C86DZB 11292119 Ki = 5720 nM T94033 CFA4O5 11293438 Ki = 2.3 nM T94033 C2WG5Z 11295972 Ki > 25000 nM T94033 CL79GU 11303092 IC50 > 10000 nM T94033 CX2UM5 11306452 Ki = 2.1 nM T94033 C2B9ZW 11306453 Ki = 0.98 nM T94033 CNCL81 11306615 Ki > 25000 nM T94033 CL2GZ0 11306789 IC50 > 10000 nM T94033 CQ5SH3 11307143 Ki = 410000 nM T94033 C72IDM 11307246 Ki > 25000 nM T94033 C0TUI9 11307532 Ki = 6500 nM T94033 CF9RM8 11307929 Ki > 25000 nM T94033 CPTV52 11316448 Ki = 12 nM T94033 C5XM9U 11317308 Ki = 0.44 nM T94033 C91GMZ 11317532 Ki = 0.4 nM T94033 CNWJ60 11318991 IC50 > 100000 nM T94033 C7ZS2B 11320069 Ki = 900 nM T94033 CVG3R6 11328459 Ki = 3.2 nM T94033 CTXB71 11329441 IC50 > 10000 nM T94033 CVAI21 11330048 Ki > 21000 nM T94033 C7EKF5 11331068 Ki = 400 nM T94033 CJI8G5 11340774 IC50 > 10000 nM T94033 C64EOX 11341794 Ki > 21000 nM T94033 CF6P9W 11342482 Ki = 1.3 nM T94033 C6CDN3 11347670 Ki = 43700 nM T94033 CLY5G8 11350400 Ki = 5310 nM T94033 CR8NW9 11351302 Ki = 8871 nM T94033 C4SCD9 11351875 Ki = 1.8 nM T94033 C8AS1B 11352537 Ki = 4.2 nM T94033 CSIM71 11353123 Ki > 25000 nM T94033 CTJ1Z2 11361949 Ki = 10160 nM T94033 C1V5ES 11363818 IC50 > 10000 nM T94033 CQ9BZ3 11363906 Ki > 25000 nM T94033 CK51RW 11364032 Ki > 25000 nM T94033 CT83NF 11364269 Ki > 25000 nM T94033 CTB9G7 11364882 Ki = 1600 nM T94033 CBT73W 11365338 Ki = 99 nM T94033 CY58QO 11365611 Ki = 0.00065 nM T94033 CBU78I 11373015 IC50 > 10000 nM T94033 C15DOY 11374307 Ki = 10 nM T94033 C4U9OQ 11374975 IC50 > 10000 nM T94033 C52YOA 11375433 IC50 > 10000 nM T94033 C9W5IX 11376076 IC50 = 63000 nM T94033 C6V5IL 11376816 Ki = 2 nM T94033 CIWL90 11386810 Ki > 25000 nM T94033 CRO4M9 11386863 Ki = 210 nM T94033 C8URO7 11387451 Ki = 15000 nM T94033 C6U5OI 11387989 Ki > 21000 nM T94033 CK1N2O 11396906 IC50 = 42 nM T94033 CZT2D7 11397246 Ki = 0.57 nM T94033 CG87TQ 11398046 IC50 > 100000 nM T94033 CR9Q3O 11399867 IC50 = 1400 nM T94033 C3DQ7J 11409073 IC50 > 10000 nM T94033 CE2NF4 11410953 Ki = 16 nM T94033 C8WZ0P 11416498 Ki = 50700 nM T94033 CVQ7G6 11419529 Ki = 2.9 nM T94033 CODR29 11420832 Ki = 45 nM T94033 CUHD35 11421628 Ki > 21000 nM T94033 CSD74B 11421657 Ki = 2100 nM T94033 C3RF5J 11433298 Ki = 0.78 nM T94033 CLH6X5 11433511 Ki = 1700 nM T94033 CCPU80 11434124 Ki > 21000 nM T94033 CN46CG 11441985 IC50 > 10000 nM T94033 C9GPF0 11444427 Ki 430 nM T94033 C2AC1M 11444632 Ki = 0.99 nM T94033 CIQH43 11445130 IC50 = 250000 nM T94033 CM7DK5 11445304 Ki = 2300 nM T94033 C9O4NF 11450922 IC50 > 62000 nM T94033 CFL61Z 11454667 Ki > 13000 nM T94033 CB60QJ 11455408 Ki > 25000 nM T94033 C2OLI9 11465119 Ki = 1.3 nM T94033 CG8H7N 11465140 IC50 > 10000 nM T94033 C8KJ1G 11466928 Ki > 21000 nM T94033 CU9LH8 11466995 IC50 > 10000 nM T94033 C0T6CN 11467119 Ki > 21000 nM T94033 CH4V9C 11468062 Ki = 740 nM T94033 CJ6TL8 11468217 Ki = 900 nM T94033 C63LIR 11473486 Ki = 3490 nM T94033 CD31BU 11478099 IC50 > 10000 nM T94033 CU04WZ 11478333 Ki = 14000 nM T94033 CVI82D 11479420 Ki = 6300 nM T94033 C5WV3Z 11489877 IC50 > 100000 nM T94033 C50FQZ 11489885 Ki = 14900 nM T94033 CNV5Q0 11491382 IC50 = 13 nM T94033 C13KMF 11510856 Ki = 1 nM T94033 CJZ09N 11512593 Ki = 2500 nM T94033 C28BMR 11513105 Ki = 420 nM T94033 CLT1I0 11518907 Ki = 349 nM T94033 CKN8R7 11525275 IC50 > 10000 nM T94033 CRNU10 11534959 Ki = 2500 nM T94033 C9M6JZ 11538422 Ki = 4700 nM T94033 C6D9FR 11540759 Ki = 5600 nM T94033 CD1A6T 11542037 Ki = 4200 nM T94033 CA8KD7 11542038 Ki = 620 nM T94033 C3USR9 11543714 IC50 > 5000 nM T94033 CBP69L 11557024 Ki = 6000 nM T94033 CCG84F 11563457 Ki = 120 nM T94033 CV46NL 11563632 Ki = 3000 nM T94033 C9UNG3 11567163 IC50 = 103 nM T94033 CU8S4Q 11568602 Ki = 2300 nM T94033 CEAZ46 11569930 Ki = 600 nM T94033 C3TJ7M 11570580 Ki = 51 nM T94033 C6RHD8 11570700 Ki = 4000 nM T94033 C1DN2L 11570759 Ki = 1500 nM T94033 C17OJS 11572844 IC50 > 5000 nM T94033 C6FG8V 11577055 Ki = 210 nM T94033 C7IG5Z 11577871 IC50 = 1.4 nM T94033 CIY34V 11577968 Ki = 260 nM T94033 CJ38EP 11577970 Ki = 200 nM T94033 C7MF9N 11578158 Ki = 300 nM T94033 CTSK74 11584729 Ki = 27000 nM T94033 C1RQ6P 11592130 Ki = 21000 nM T94033 CBC84M 11592593 Ki = 9400 nM T94033 C7ZS8L 11592600 Ki = 460 nM T94033 CFJR86 11600024 IC50 = 500 nM T94033 C7QTY8 11606981 Ki = 4000 nM T94033 CU07NO 11607091 Ki = 5400 nM T94033 CL9TZ2 11614477 Ki = 20000 nM T94033 C1R2WJ 11618823 Ki = 8 nM T94033 CB4O2Q 11621579 Ki = 1300 nM T94033 CD3R1E 11627899 Ki = 7000 nM T94033 CB9P0Q 11628768 Ki = 1800 nM T94033 C6UAV3 11632008 IC50 > 5000 nM T94033 CO3Q9N 11635973 Ki = 1200 nM T94033 CRX98P 11636026 Ki = 1800 nM T94033 C91JNO 11639020 IC50 > 5000 nM T94033 CW10CL 11642802 Ki = 1800 nM T94033 C4MCW2 11646889 IC50 > 5000 nM T94033 C1O5ZV 11648797 Ki = 149 nM T94033 CH20JE 11652994 IC50 > 5000 nM T94033 C2W5XF 11656797 Ki = 8800 nM T94033 C4SAR0 11657278 Ki = 54 nM T94033 CFM4V3 11663836 IC50 = 17 nM T94033 CVQ16C 11664107 Ki = 170 nM T94033 CPZG49 11664334 Ki = 2600 nM T94033 CT9E0G 11664643 Ki = 1600 nM T94033 CWV87X 11671266 Ki = 13000 nM T94033 CE0A6N 11671776 Ki = 490 nM T94033 C85GCY 11671956 Ki = 5000 nM T94033 C1DHO6 11678360 Ki = 12000 nM T94033 C4IBO3 11678764 Ki = 99 nM T94033 CJP9O1 11684611 Ki > 12610 nM T94033 C69YSR 11693028 Ki = 16000 nM T94033 CCQY30 11693049 Ki = 420 nM T94033 CPFW75 11699600 Ki = 190 nM T94033 C3VS2H 11699903 Ki = 270 nM T94033 CNV09Z 11699913 Ki = 210 nM T94033 C5Z6YE 11700643 Ki = 7300 nM T94033 CKQ4O2 11721188 Ki = 1400 nM T94033 C4UB2X 11721375 Ki = 580 nM T94033 C4M0XP 11725377 IC50 = 100000 nM T94033 CGA9V3 11725721 Ki = 26 nM T94033 CJZA24 11729069 Ki > 5000 nM T94033 C9SW2I 11729577 IC50 = 20400 nM T94033 CL4CN3 11729890 Ki = 4200 nM T94033 CCI97J 11730048 IC50 = 3000 nM T94033 CS12RM 11730232 Ki = 3900 nM T94033 CBJ4R6 11730277 Ki > 21000 nM T94033 CGJ32L 11730366 IC50 = 106000 nM T94033 CI2KC5 11730368 Ki = 1230 nM T94033 CA12MJ 11730381 IC50 = 260 nM T94033 C7D1KA 11730408 IC50 = 260 nM T94033 CQ0ZP6 11730472 Ki > 3900 nM T94033 CN0HF5 11730512 IC50 > 100000 nM T94033 C7D8HR 11731179 Ki = 1180 nM T94033 CCYI90 11731292 IC50 = 1000 nM T94033 C86CXE 11732210 IC50 = 33000 nM T94033 C8K1ZJ 11733007 Ki > 5000 nM T94033 CAF10R 11733131 IC50 > 30000 nM T94033 CN6X4B 11733626 Ki = 44 nM T94033 CCKF59 11733750 IC50 > 30000 nM T94033 CC3E2I 11733884 IC50 = 37700 nM T94033 CH17KD 11734055 IC50 = 9150 nM T94033 C7LW3O 11734113 Ki = 57000 nM T94033 CF0L9M 11734243 Ki = 15 nM T94033 CO8P4U 11734268 IC50 > 30000 nM T94033 CQ5U8H 11739438 Ki = 6920 nM T94033 CLOA31 11740543 Ki = 125 nM T94033 CNZ04Q 11740591 Ki = 1.5 nM T94033 C6SZX7 11741904 Ki = 480 nM T94033 CR53AD 11742672 Ki = 15 nM T94033 C8QZK0 11743193 Ki > 5000 nM T94033 C5VN3J 11744466 Ki = 2 nM T94033 CM95SZ 11744578 IC50 = 3190 nM T94033 C4LMF0 11751278 Ki = 9 nM T94033 CX18BY 11752965 Ki > 21000 nM T94033 CP3FI1 11753847 Ki = 160 nM T94033 CIMG42 11754250 Ki = 18.3 nM T94033 C1LPF4 11754261 IC50 > 10000 nM T94033 CZ2W6F 11754502 Ki = 210 nM T94033 CAI6P1 11754992 Ki = 200 nM T94033 CNPW05 11755188 IC50 > 10000 nM T94033 C5VXD6 11755549 Ki < 0.01 nM T94033 CUMO51 11756555 IC50 > 10000 nM T94033 CS0JR2 11756961 Ki = 2900 nM T94033 C84BVH 11757010 Ki = 1 nM T94033 C83GXL 11757017 IC50 = 530 nM T94033 CT7EI2 11757135 Ki = 9000 nM T94033 CGJ80T 11758070 Ki = 6.7 nM T94033 CMR6A0 11758260 Ki > 13000 nM T94033 C95TSZ 11758428 Ki = 0.7 nM T94033 C7P4CG 11758475 Ki > 13000 nM T94033 CU9D5M 11760897 IC50 = 4600 nM T94033 CG82LK 11761121 Ki > 5000 nM T94033 CZ7QI3 11761613 Ki > 5000 nM T94033 C07WYX 11762017 Ki = 0.1 nM T94033 C5H7AR 11762101 IC50 = 4000 nM T94033 CJVR18 11762113 Ki > 2100 nM T94033 C4F0HE 11762405 Ki = 0.9 nM T94033 CZ34HE 11762589 IC50 = 150 nM T94033 CZ91LI 11762766 Ki = 770 nM T94033 CV9BN2 11762839 IC50 = 7630 nM T94033 C7JLR1 11774107 Ki = 21700 nM T94033 CR2E9T 11782463 Ki = 120 nM T94033 C9LC5W 11784323 Ki > 5000 nM T94033 CMH70L 11784384 Ki = 56 nM T94033 C1BIN4 11785755 Ki = 3900 nM T94033 CN3IG5 11785929 Ki > 25000 nM T94033 CR5W1D 11785966 Ki = 3700 nM T94033 C7Z4MV 11785967 IC50 = 58000 nM T94033 CK4CH2 11786303 Ki > 25000 nM T94033 CU9RW5 11792439 Ki > 21000 nM T94033 CT0MA8 11793538 IC50 = 1320 nM T94033 C8LD7W 11793807 Ki = 2900 nM T94033 C4SLV5 11794918 Ki = 2.5 nM T94033 CAGC25 11795137 Ki = 2600 nM T94033 C83DOK 11796018 IC50 = 5 nM T94033 CZ62LI 11796080 Ki = 730 nM T94033 CP2I9G 11796404 Ki = 0.52 nM T94033 CW6DG1 11796805 Ki > 5000 nM T94033 CF1S2R 11796942 Ki = 3300 nM T94033 CT97QL 11797044 IC50 = 50 nM T94033 C8EHN3 11797101 Ki = 24 nM T94033 CIS51A 11797515 Ki = 12 nM T94033 CZM62X 11797951 Ki = 2040 nM T94033 CH2Z1N 11798267 Ki = 21000 nM T94033 CK8MI3 11798429 Ki = 3700 nM T94033 CA6SL9 11799353 Ki = 85 nM T94033 CTOK74 11799409 Ki = 54 nM T94033 C2HS4G 11800433 Ki = 3.8 nM T94033 CK31IT 11800766 Ki = 360 nM T94033 CL6Z3G 11801417 Ki = 2.2 nM T94033 C68VNG 11801427 Ki = 1800 nM T94033 CL01GT 11801580 Ki = 5800 nM T94033 CVZ82O 11801725 Ki = 2700 nM T94033 CFP36D 11802531 Ki = 4000 nM T94033 CY46UZ 11802721 Ki = 13000 nM T94033 CPJS89 11811066 Ki = 63 nM T94033 CO5X8E 11811735 Ki = 15 nM T94033 C5HL6W 11811831 IC50 = 270 nM T94033 CL0W8P 11812192 Ki = 32 nM T94033 CG7HY3 11812211 IC50 = 11300 nM T94033 CPR54N 11812296 Ki = 0.042 nM T94033 CZIB40 11812370 Ki = 1.3 nM T94033 CI9AM0 11812634 IC50 = 20000 nM T94033 C4XE8C 11812643 Ki = 16 nM T94033 CIL1Z6 11813042 Ki = 0.29 nM T94033 C1IY9C 11813203 IC50 = 2100 nM T94033 C9VW2P 11813305 Ki > 3900 nM T94033 CDQC29 11813421 IC50 = 890 nM T94033 CTUV60 11813618 IC50 < 40 nM T94033 CA6BQ4 11813669 IC50 > 100000 nM T94033 C1UQ6O 11813975 Ki = 13500 nM T94033 C8INH6 11814686 IC50 = 11200 nM T94033 C98ZOR 11824040 Ki = 22000 nM T94033 CYX74A 11824584 Ki = 65000 nM T94033 CCT84E 11825785 Ki > 5000 nM T94033 CEYP62 11826299 Ki = 99000 nM T94033 C8ON2Z 11826539 IC50 = 28400 nM T94033 C3EFY7 11826875 Ki > 21000 nM T94033 CIO26S 11826929 Ki = 16 nM T94033 C3AP8E 11826975 IC50 = 4740 nM T94033 C7LUI9 11827030 IC50 > 30000 nM T94033 C93TLO 11827247 Ki = 3290 nM T94033 CIR2M0 11827276 IC50 = 2890 nM T94033 C0A8LS 11827475 IC50 = 5200 nM T94033 C63PXR 11827585 Ki = 0.17 nM T94033 CE5US8 11827739 IC50 = 2100 nM T94033 C61GPA 11828451 IC50 = 60000 nM T94033 CW6E7I 11828640 IC50 > 30000 nM T94033 CC6M2W 11849330 IC50 > 33000 nM T94033 C1T6CS 11849331 IC50 = 100000 nM T94033 CRT0N2 11849332 IC50 = 33000 nM T94033 C21OSF 11849333 IC50 = 300000 nM T94033 CLH9U6 11849334 IC50 = 300000 nM T94033 CGB6W0 11849371 IC50 > 33000 nM T94033 CX5BV1 11849373 IC50 = 10050 nM T94033 CH7BM8 11849374 IC50 > 300000 nM T94033 C0K7UZ 11849375 IC50 = 4400 nM T94033 CPR12Z 11849376 IC50 > 33000 nM T94033 C82FJL 11849424 IC50 = 300000 nM T94033 C89XNT 11849425 IC50 = 100000 nM T94033 C8TVZ9 11849426 IC50 = 770 nM T94033 CF7UX3 11849427 IC50 > 300000 nM T94033 CW1QF2 11849428 IC50 > 300000 nM T94033 CEO7G0 11849429 IC50 > 300000 nM T94033 CR5H3J 11849462 IC50 > 33000 nM T94033 C1JBR8 11849463 IC50 = 13340 nM T94033 C56NRA 11957383 IC50 = 1200 nM T94033 CNS8I9 11963488 IC50 = 20.2 nM T94033 CJ02OR 11963489 IC50 = 47.3 nM T94033 C5SEB3 11967063 IC50 > 30000 nM T94033 CTB2C9 11967128 IC50 = 3190 nM T94033 C0MCS3 11979744 IC50 = 18 nM T94033 C69HNO 11984565 Ki = 13000 nM T94033 CL50RW 12010538 Ki = 654 nM T94033 CI48TS 12010539 Ki = 119 nM T94033 C5D0IW 12017717 Ki = 79 nM T94033 CCHL86 12017718 Ki = 1180 nM T94033 CX8W6S 12017719 Ki = 240 nM T94033 C69DQA 12017720 Ki = 350 nM T94033 CK1BX3 12017721 Ki = 93 nM T94033 CE84MP 12017722 Ki = 38 nM T94033 CK16XW 12017723 Ki = 56 nM T94033 CC93ZQ 12017724 Ki = 52 nM T94033 CFWM35 12017725 Ki = 24 nM T94033 C4CL6P 12017726 Ki = 65 nM T94033 CHT3M8 12017727 Ki = 182 nM T94033 CTA80I 12017728 Ki = 1000 nM T94033 CK5UB4 12017729 Ki = 38320 nM T94033 C1K4FT 12017730 Ki = 7830 nM T94033 C2EF8D 12041284 IC50 = 9.5 nM T94033 C6UT2G 12042266 Ki = 1.6 nM T94033 CQG4D9 12042267 Ki = 0.33 nM T94033 CBL13C 12042268 Ki = 36 nM T94033 C7OC2I 12042269 Ki = 0.36 nM T94033 C4J2IX 12042961 IC50 = 670 nM T94033 CPR4I1 12047383 Ki = 126 nM T94033 C5U0FJ 12047384 Ki = 280 nM T94033 C5FU3H 12047385 Ki = 118 nM T94033 CP3Q4D 12052450 Ki = 5 nM T94033 CX98PQ 12082573 IC50 > 1000000 nM T94033 CT7IR8 12110710 IC50 = 6000 nM T94033 CJL46R 12254250 Ki = 398107.17 nM T94033 C5PVL9 12456162 Ki = 2511886.43 nM T94033 CS7F2T 12967905 Ki = 6.3 nM T94033 C05YMF 12967907 Ki = 1.2 nM T94033 C84CJL 12986348 IC50 > 10000 nM T94033 CTUN59 12991294 Ki = 6.8 nM T94033 CG4W6K 15021502 IC50 = 7500 nM T94033 CP35QH 15227625 Ki = 7000 nM T94033 CBVA60 15227963 Ki = 631 nM T94033 CFO06N 15227964 Ki = 316 nM T94033 CB91UM 15227967 Ki = 23 nM T94033 CG2L9I 15228005 Ki = 1585 nM T94033 C24DXU 15285659 Ki = 0.46 nM T94033 CZ6TK8 15289347 Ki = 240000 nM T94033 C8JC1A 15295705 Ki = 3.3 nM T94033 CB1I0K 15295707 Ki = 26 nM T94033 C8KPA4 15295709 Ki = 4.3 nM T94033 CVG34T 15295712 Ki = 0.4 nM T94033 C60TVD 15392306 IC50 > 10000 nM T94033 C3HYW7 15431805 IC50 = 0.57 nM T94033 CIE47P 15434242 Ki = 1.8 nM T94033 CZBD56 15435386 Ki = 16000 nM T94033 CY42MO 15449319 IC50 = 73 nM T94033 CFJB64 15449320 IC50 = 92 nM T94033 C48WFU 15449321 IC50 = 98 nM T94033 CGX57Z 15454127 Ki = 350 nM T94033 CKH1S3 15458385 Ki = 0.2 nM T94033 C9KJ5Y 15461560 Ki = 800 nM T94033 CM2RN1 15461564 Ki = 40 nM T94033 CSHJ59 15462938 Ki = 24 nM T94033 CBYG78 15462942 Ki = 24 nM T94033 CIA8P9 15487292 IC50 = 11200 nM T94033 CX5S1Z 15511974 Ki = 900 nM T94033 CW2QY0 15515689 IC50 = 160 nM T94033 CG9Q0P 15515690 IC50 = 120 nM T94033 C54SUM 15515691 IC50 = 220 nM T94033 CMR59D 15515698 Ki = 40 nM T94033 C4LXI5 15515699 Ki = 2500 nM T94033 C6Y8UK 15515700 Ki = 3000 nM T94033 C5EA6G 15515701 Ki = 290 nM T94033 C9JKS1 15515702 Ki = 3500 nM T94033 CKGJ08 15516769 IC50 = 880 nM T94033 C5Z4MG 15516770 Ki = 55 nM T94033 C3YR6T 15516779 IC50 = 110 nM T94033 C58YJC 15518434 Ki = 2 nM T94033 CD8F0P 15518435 Ki = 5.5 nM T94033 CL64JN 15518436 Ki = 0.1 nM T94033 CZMK79 15518437 Ki = 0.5 nM T94033 C7V6RN 15518438 Ki = 0.06 nM T94033 CGQ09C 15519903 Ki = 36 nM T94033 CKH64M 15519904 Ki = 49890 nM T94033 CZ57HV 15519905 Ki = 1800 nM T94033 CQ0M5U 15519907 Ki = 100 nM T94033 CINA41 15519912 Ki = 12 nM T94033 C60JFG 15521694 Ki = 10100 nM T94033 CP63GF 15534822 IC50 = 17.9 nM T94033 CPJT95 15545832 Ki = 1350 nM T94033 C0DQ2E 15546243 Ki = 1500000 nM T94033 CN6M4K 15858923 Ki = 990 nM T94033 CN97QO 15858924 Ki = 9.4 nM T94033 CZ56MD 15858926 Ki = 9.1 nM T94033 CL9T7Y 15870100 Ki = 11000 nM T94033 CB3T9P 15870101 Ki = 7300 nM T94033 C9EH2Y 15887336 Ki = 4 nM T94033 CT12GL 15895095 Ki = 1300 nM T94033 CF7KG1 15908935 Ki = 5500 nM T94033 CK6MH4 15908936 Ki = 5400 nM T94033 CW73FT 15923398 Ki = 125 nM T94033 C6VZ1N 15942655 Ki = 71500 nM T94033 CL93AK 15946227 IC50 = 4400 nM T94033 CA86KZ 15947513 Ki = 8700 nM T94033 CU0O5N 15947601 Ki = 7800 nM T94033 CQ3RF8 15947602 Ki = 7900 nM T94033 CS8HY6 15947811 Ki = 9500 nM T94033 CCMQ45 15947923 Ki = 6700 nM T94033 CUGI75 15947926 Ki = 11000 nM T94033 CSV70B 15948627 Ki = 12000 nM T94033 CSAU78 15949836 IC50 = 1980 nM T94033 C7VH6K 15950345 Ki = 400 nM T94033 C2QO1B 15955412 Ki > 50000 nM T94033 C19ARJ 15984063 Ki = 64000 nM T94033 CLP2D3 16004672 Ki = 170 nM T94033 CA8Y1K 16046152 Ki = 305 nM T94033 CNBJ60 16046153 Ki = 245 nM T94033 C5TBL6 16049247 IC50 = 17000 nM T94033 CC7Y0D 16066741 IC50 > 200000 nM T94033 C9BH4X 16086308 IC50 = 4900 nM T94033 CF1V2N 16086310 IC50 = 22000 nM T94033 C9JX7U 16086312 IC50 = 4300 nM T94033 CK7IM0 16086316 IC50 = 7500 nM T94033 CT9QM5 16086318 IC50 = 34000 nM T94033 CXO65R 16086320 IC50 = 6300 nM T94033 C3EUJ6 16086336 IC50 = 770 nM T94033 CR9EN3 16086338 IC50 = 6000 nM T94033 CR7B3D 16086340 IC50 = 35000 nM T94033 C90CXM 16086342 IC50 = 1670 nM T94033 C7T5AI 16086344 IC50 = 2980 nM T94033 CJZ63N 16086346 IC50 = 67000 nM T94033 C05XAN 16086348 IC50 = 15900 nM T94033 CACN42 16086349 IC50 = 1500 nM T94033 CDSM46 16098887 IC50 = 6700 nM T94033 CFK98M 16098895 IC50 = 1000 nM T94033 C6BQ0G 16098896 IC50 = 7700 nM T94033 C1ZXL4 16098897 IC50 = 27000 nM T94033 CP6Y7Q 16098898 IC50 = 10000 nM T94033 C3J6LO 16098899 IC50 = 12000 nM T94033 CQ4YJ8 16098900 IC50 = 1400 nM T94033 CDL2X5 16098901 IC50 = 390 nM T94033 C53ZXO 16098902 IC50 = 3100 nM T94033 CUJ5A9 16098903 IC50 = 2800 nM T94033 CZ3WM4 16098905 IC50 > 200000 nM T94033 CVN8Y1 16098906 IC50 = 976 nM T94033 CTY5W9 16098907 IC50 = 5600 nM T94033 CSBT08 16098908 IC50 = 523 nM T94033 CR9DT0 16098909 IC50 = 606 nM T94033 C53YRO 16098910 IC50 = 2040 nM T94033 C91CQM 16098911 IC50 = 440 nM T94033 C0W5NR 16098912 IC50 = 400 nM T94033 CS21OE 16098913 IC50 = 710 nM T94033 CTR91H 16111809 Ki = 700 nM T94033 CYKU84 16111812 Ki = 1500 nM T94033 CPKT43 16111813 Ki = 400 nM T94033 C24FJO 16111815 Ki = 5400 nM T94033 C08LZU 16111821 Ki = 4400 nM T94033 CG95BH 16111822 Ki = 1200 nM T94033 C3FOW4 16111824 Ki = 5300 nM T94033 CYTJ73 16111827 Ki = 3700 nM T94033 COJI93 16111856 Ki = 900 nM T94033 CFZ8N2 16111857 Ki = 900 nM T94033 C0K6MZ 16111859 Ki = 6400 nM T94033 CQ8MJ5 16111860 Ki = 2500 nM T94033 C8C7IP 16111861 Ki = 1000 nM T94033 CJP3Q0 16111862 Ki = 1000 nM T94033 CY95DW 16111863 Ki = 2500 nM T94033 CF5BU9 16111864 Ki = 8000 nM T94033 C6BFU3 16111865 Ki = 11500 nM T94033 C9OSM6 16144480 Ki > 15000 nM T94033 CDR0G7 16145606 Ki = 1700 nM T94033 CY20PW 16147332 Ki = 750 nM T94033 CF5Y3L 16147570 Ki > 15000 nM T94033 C7S6IT 16148231 Ki > 15000 nM T94033 C0R4PG 16214382 IC50 = 130000 nM T94033 CA0Y5E 16219042 Ki = 1000000 nM T94033 CN6CJ2 16220264 IC50 = 56100 nM T94033 CZ7FS4 16284785 IC50 > 200000 nM T94033 C56TPZ 16285203 IC50 > 200000 nM T94033 C1KZB9 16289649 IC50 > 200000 nM T94033 CPK67M 16664096 Ki = 1200 nM T94033 CU60AH 16718671 IC50 = 32200 nM T94033 COAB94 16718712 IC50 = 3800 nM T94033 CU28CE 16718713 IC50 = 1130 nM T94033 CLI4D7 16718757 IC50 = 2350 nM T94033 C2SFC0 16718759 IC50 = 20000 nM T94033 CC20PS 16718760 IC50 = 125000 nM T94033 CCKO80 16718762 IC50 = 8100 nM T94033 C37MRI 16718808 IC50 = 2400 nM T94033 CJL72U 16731819 Ki = 1300 nM T94033 C05JSB 16731821 Ki = 1500 nM T94033 C6SN2Q 16731823 Ki = 680 nM T94033 CG49VM 16731824 Ki > 5000 nM T94033 C8ZFY6 16731827 Ki = 2600 nM T94033 CN60KL 16731975 Ki = 5400 nM T94033 CB01OR 16731976 Ki = 1700 nM T94033 C7MR9E 16731977 Ki = 1400 nM T94033 CF4V3D 16731978 Ki = 1400 nM T94033 CS2QJ8 16731979 Ki = 770 nM T94033 CYB1E0 16731980 Ki = 1400 nM T94033 CD64LP 16732121 Ki = 1100 nM T94033 CWU9D7 16732123 Ki = 2100 nM T94033 CH2U5Z 16732125 Ki = 1100 nM T94033 CSB43R 16732126 Ki = 1200 nM T94033 CK74UL 16732127 Ki = 300 nM T94033 C4A1RO 16732128 Ki = 190 nM T94033 C9BD4C 16732263 Ki = 340 nM T94033 CZ3M6S 16732265 Ki = 340 nM T94033 C3DW7C 16732266 Ki = 450 nM T94033 CBO97E 16732268 Ki = 360 nM T94033 C7QBR0 16732402 Ki = 140 nM T94033 C6RPF4 16732404 Ki = 630 nM T94033 CN3D9T 16732406 Ki = 470 nM T94033 C1HFQ6 16732407 Ki > 5000 nM T94033 CGC0Q2 16732555 Ki = 1700 nM T94033 C7SUK0 16732557 Ki = 2000 nM T94033 CT4K0V 16732559 Ki = 410 nM T94033 CKAZ40 16732560 Ki = 580 nM T94033 CKN73Z 16732562 Ki = 160 nM T94033 CLF90N 16732707 Ki = 90 nM T94033 CR3K2E 16732708 Ki = 100 nM T94033 C2EOR6 16732711 Ki = 970 nM T94033 CPK8Z7 16732713 Ki = 1100 nM T94033 CUHT92 16732866 Ki = 2600 nM T94033 C07OPV 16732868 Ki = 1500 nM T94033 C3Y2HE 16732871 Ki = 2200 nM T94033 C47UEZ 16732873 Ki = 3300 nM T94033 CL4EW1 16733006 Ki = 3300 nM T94033 CNYA03 16733007 Ki = 920 nM T94033 C7XU2R 16733008 Ki = 630 nM T94033 CRBI26 16733010 Ki = 510 nM T94033 CUEL18 16733012 Ki = 440 nM T94033 C6OK0W 16733013 Ki = 3500 nM T94033 C0G7KW 16733150 Ki = 860 nM T94033 C87WGF 17750368 Ki > 500000 nM T94033 CVY8D6 17753625 IC50 = 1.6 nM T94033 C2K9GC 17788740 Ki = 440000 nM T94033 CVB82P 17809181 IC50 = 64 nM T94033 CB6R1Z 17809213 IC50 = 14.87 nM T94033 C9PVW1 17822583 Ki > 10000 nM T94033 C5RSD3 18318130 Ki = 400 nM T94033 CL13IP 18318139 Ki = 3260 nM T94033 C3P0VK 18318146 Ki = 480 nM T94033 COJ9F3 18318187 Ki = 1000 nM T94033 C1S3MX 18318188 Ki = 2140 nM T94033 CGNJ35 18318198 Ki = 5000 nM T94033 CE7RZ4 18318201 Ki = 4700 nM T94033 CBS40I 18318220 Ki = 2900 nM T94033 CC8K3N 18322173 Ki = 1600 nM T94033 CFL1O5 18322175 Ki = 640 nM T94033 CYL61S 18322190 Ki = 7620 nM T94033 C97AVH 18322194 Ki = 2900000 nM T94033 CV0NH9 18322205 Ki = 880 nM T94033 CI5J3Y 18376546 Ki > 5000 nM T94033 CMU9A3 18376555 Ki > 5000 nM T94033 CFQE53 18376558 Ki > 5000 nM T94033 CLUC36 18376562 Ki = 2300 nM T94033 C76KJP 18376565 Ki > 5000 nM T94033 CC94AD 18376598 Ki > 5000 nM T94033 CJ7K3O 18376605 Ki = 1500 nM T94033 C1UT4K 18376606 Ki > 5000 nM T94033 CU98XE 18376618 Ki = 1000 nM T94033 CCH92J 18376625 Ki > 5000 nM T94033 C25PXL 18376627 Ki > 5000 nM T94033 CL4UC9 18376641 Ki = 1100 nM T94033 C4TCP6 18376642 Ki = 190 nM T94033 C0D1EH 18376656 Ki = 4400 nM T94033 CN8CI1 18376659 Ki = 4400 nM T94033 CTA57Y 18376663 Ki = 3600 nM T94033 CHO4P2 18376665 Ki > 5000 nM T94033 CPGX36 18376669 Ki = 830 nM T94033 CG0N9Q 18376671 Ki > 5000 nM T94033 CU7V4F 18376679 Ki > 5000 nM T94033 CIJG48 18376696 Ki > 5000 nM T94033 C27NVA 18376714 Ki = 3300 nM T94033 CR1C3F 18376717 Ki > 5000 nM T94033 CSJZ89 18376719 Ki = 120 nM T94033 CUE92D 18376730 Ki > 5000 nM T94033 CPT6W5 18376743 Ki > 5000 nM T94033 CZ7HJ6 18376748 Ki > 5000 nM T94033 CXW37R 18376768 Ki > 5000 nM T94033 CBO4I0 18376780 Ki > 5000 nM T94033 C7JF8K 18376782 Ki > 5000 nM T94033 C86WAR 18376800 Ki > 5000 nM T94033 CUZ8V3 18376816 Ki > 5000 nM T94033 CAQ7X0 18376821 Ki > 5000 nM T94033 C7Y8FD 18376826 Ki > 5000 nM T94033 CRA3Y5 18376827 Ki = 510 nM T94033 C4I9XE 18376832 Ki = 160 nM T94033 C0S9XW 18376837 Ki > 5000 nM T94033 CG98XS 18376838 Ki > 5000 nM T94033 C4JE8S 18376839 Ki > 5000 nM T94033 CN1ZX0 18376843 Ki = 550 nM T94033 C8YF1V 18376848 Ki > 5000 nM T94033 CS79AF 18376858 Ki > 5000 nM T94033 C9FDM4 18376865 Ki > 5000 nM T94033 CUIC43 18376871 Ki > 5000 nM T94033 CJL9E5 18376880 Ki = 990 nM T94033 C8KTW9 18376881 Ki > 5000 nM T94033 C63EFY 18376882 Ki = 2700 nM T94033 CE2BH4 18376888 Ki = 1000 nM T94033 CE43LC 18376891 Ki > 5000 nM T94033 C9V3HX 18376897 Ki > 5000 nM T94033 C1ZKY8 18376901 Ki > 5000 nM T94033 CH8R6S 18376905 Ki = 310 nM T94033 CUJP51 18376916 Ki > 5000 nM T94033 CLE27U 18376919 Ki = 1500 nM T94033 C3EN2U 18376921 Ki = 1800 nM T94033 CM6NT1 18376930 Ki = 560 nM T94033 CG8Y0C 18376939 Ki = 2300 nM T94033 C1SZ9Q 18376940 Ki > 5000 nM T94033 CWG72T 18376950 Ki > 5000 nM T94033 CV3ZE2 18376959 Ki > 5000 nM T94033 CWI0E3 18376970 Ki > 5000 nM T94033 C1OM7T 18376973 Ki = 160 nM T94033 C1T3VP 18376976 Ki = 2400 nM T94033 C7SO8U 18376989 Ki > 5000 nM T94033 CF0GR6 18376995 Ki > 5000 nM T94033 CN2JE5 18376999 Ki > 5000 nM T94033 CC9ZE2 18377002 Ki = 1000 nM T94033 C53XHD 18377003 Ki > 5000 nM T94033 C94LUS 18377010 Ki > 5000 nM T94033 C79ZIE 18377020 Ki > 5000 nM T94033 C3FYR1 18377031 Ki > 5000 nM T94033 CI5U7D 18377033 Ki > 5000 nM T94033 CEH2K1 18377041 Ki > 5000 nM T94033 CX8RE3 18377048 Ki > 5000 nM T94033 CTQ85L 18397340 Ki > 1000000 nM T94033 CZ4L5C 18397341 Ki = 130000 nM T94033 CU5N8E 18397342 Ki = 112000 nM T94033 C4HE7G 18397344 Ki = 36000 nM T94033 CF1Y7P 18397345 Ki = 213000 nM T94033 C3D1VS 18397346 Ki = 29000 nM T94033 CEJ3K1 18397347 Ki = 537000 nM T94033 CVB47A 18397350 Ki > 1000000 nM T94033 C7DB0W 18397352 Ki = 59500 nM T94033 C03OYT 18397353 Ki > 1000000 nM T94033 CP3ZL0 18397354 Ki > 1000000 nM T94033 CM28UY 18397357 Ki = 255000 nM T94033 C0POA1 18397359 Ki > 1000000 nM T94033 CSW0L3 18397360 Ki > 1000000 nM T94033 CN9S6X 18397370 Ki > 1000000 nM T94033 CS21RN 18397380 Ki = 146000 nM T94033 C7PRY3 18412330 IC50 = 3.23 nM T94033 CD4IN3 18412338 IC50 = 5.37 nM T94033 CN87FW 18474271 Ki = 99 nM T94033 C3V9EC 18549309 Ki = 400 nM T94033 CF7L0E 18657594 IC50 > 40000 nM T94033 C8IN3S 18657595 IC50 = 5500 nM T94033 CL3E1V 18657596 IC50 > 115000 nM T94033 CAW35I 18669708 Ki = 204 nM T94033 C1ERT0 18671884 Ki = 15 nM T94033 COUY03 18671891 Ki = 120 nM T94033 CXQ8G0 18671904 Ki = 47 nM T94033 C9BKU4 18671915 Ki = 13 nM T94033 CC6AT5 18671918 Ki = 66 nM T94033 CQ1JT8 18671920 Ki = 47 nM T94033 C9NB0Z 18675062 IC50 = 1100 nM T94033 C09KIY 18675079 IC50 = 910 nM T94033 C29WYS 18675086 IC50 = 890 nM T94033 CR6I5L 18675103 IC50 = 65000 nM T94033 CLZ97R 18675188 IC50 = 1700 nM T94033 CK6U1I 18675238 IC50 = 1900 nM T94033 CD9UE4 18675298 IC50 = 5600 nM T94033 CF4W5D 18727604 IC50 > 10000 nM T94033 CB0IQ4 18727607 IC50 > 11000 nM T94033 C31ZAL 18727831 IC50 > 11000 nM T94033 CJY67O 18727833 IC50 > 11000 nM T94033 C02HEA 18727834 IC50 > 11000 nM T94033 CJSL38 18727836 IC50 > 11000 nM T94033 C8AMY9 18727838 IC50 > 11000 nM T94033 CY8AC3 18727841 IC50 > 11000 nM T94033 CD02TK 18727852 IC50 > 11000 nM T94033 C1JMX5 18727855 IC50 > 11000 nM T94033 CE4PI7 18741279 Ki = 0.8 nM T94033 CNUR53 18800583 Ki = 2700 nM T94033 CMA2G0 18800591 Ki > 21000 nM T94033 CXI52J 18800605 Ki = 300 nM T94033 CYK61X 18943987 IC50 > 50000 nM T94033 CXRY67 19080908 Ki = 10 nM T94033 CAZ56G 19388089 Ki = 2800 nM T94033 C5MR0U 20585828 IC50 > 10000 nM T94033 C7P4UB 20585829 IC50 > 10000 nM T94033 CO2JG4 20595081 IC50 > 11000 nM T94033 CM7BH1 20595091 IC50 > 11000 nM T94033 CCH5N1 20595225 IC50 > 11000 nM T94033 C2ID8R 20595260 IC50 > 10000 nM T94033 CMT46A 20595328 IC50 > 10000 nM T94033 C43UDK 20608737 IC50 > 30000 nM T94033 CW3I9O 20608738 IC50 > 30000 nM T94033 C4UZO0 20608741 IC50 > 30000 nM T94033 C9Z2VH 20608755 IC50 > 30000 nM T94033 C3OF2S 20608756 IC50 > 30000 nM T94033 CMX4Q6 20608776 IC50 > 30000 nM T94033 CXH09O 20631502 IC50 = 110.48 nM T94033 CT7I1B 20641743 IC50 = 7000 nM T94033 C7LHE8 20641745 IC50 = 6000 nM T94033 CM04US 20649518 Ki = 102000 nM T94033 CTY8G2 20707887 Ki > 4000 nM T94033 C0BKY3 20707927 IC50 = 7700 nM T94033 C0FRB4 20708055 IC50 = 3800 nM T94033 CLM02X 20708056 IC50 = 5300 nM T94033 C74LUP 20708058 IC50 = 3300 nM T94033 CI6ZK4 20708066 IC50 = 4300 nM T94033 CC3I4M 20708069 IC50 = 2400 nM T94033 CJL5M6 20708073 IC50 = 2000 nM T94033 CRK8N0 20708078 IC50 = 7200 nM T94033 CC50OV 20708079 IC50 = 9000 nM T94033 C7JMO0 20708106 IC50 = 18000 nM T94033 C02MHB 20708108 IC50 = 4800 nM T94033 CL13GC 20708219 IC50 = 8700 nM T94033 CZ6KH9 20760195 Ki = 1800 nM T94033 CIM9C3 20801121 IC50 = 1790 nM T94033 CC1Y0R 20801139 IC50 = 1550 nM T94033 C4V8ZR 20801142 IC50 = 1560 nM T94033 CS3HB4 20801160 IC50 = 890 nM T94033 CGD57F 20802932 IC50 > 30000 nM T94033 CO2FM4 20802944 IC50 > 30000 nM T94033 CYUF07 20802951 IC50 = 8000 nM T94033 C1P0WC 20802959 IC50 > 30000 nM T94033 CBL6N1 20802966 IC50 > 30000 nM T94033 C27ZJT 20802995 IC50 > 100000 nM T94033 CTNW09 21125474 IC50 = 300 nM T94033 CA3P9S 21182630 Ki = 7 nM T94033 C5BVK0 21182636 Ki = 5.1 nM T94033 CLUP41 21182654 Ki = 4.1 nM T94033 CIKQ90 21182692 Ki = 5.1 nM T94033 CBI8T1 21182760 Ki = 3.8 nM T94033 CGD98Q 21182787 Ki = 0.3 nM T94033 CO37IL 21182800 Ki = 0.5 nM T94033 C8HN9Y 21182873 Ki = 7.2 nM T94033 CX28DT 21182884 Ki = 11 nM T94033 C17GNE 21182938 Ki = 0.9 nM T94033 C59JBT 21182950 Ki = 1.9 nM T94033 C23NLP 21191106 Ki = 2.3 nM T94033 C1B5UW 21217905 Ki = 400 nM T94033 CR6C2I 21218691 Ki = 16000 nM T94033 CS5L2M 21218709 Ki = 14100 nM T94033 CEQ6B2 21218732 Ki > 21000 nM T94033 C79ZNM 21218751 Ki > 21000 nM T94033 CLT36V 21250176 IC50 = 5 nM T94033 CGC48U 21250249 IC50 = 37 nM T94033 CE0T3P 21250257 IC50 = 87 nM T94033 CRYB96 21250293 IC50 = 8 nM T94033 C0ECB5 21250297 IC50 = 3300 nM T94033 CF3YS0 21250354 IC50 = 196 nM T94033 CLV49W 21250386 IC50 = 16 nM T94033 CN2YE9 21250416 IC50 = 27 nM T94033 CRD4V1 21250427 IC50 = 13 nM T94033 C3T5SA 21250434 IC50 = 68 nM T94033 C9H7ZI 21250518 IC50 = 10 nM T94033 CNTI15 21366511 IC50 > 11000 nM T94033 C5S8ZW 21366513 IC50 > 11000 nM T94033 C67QCO 21366574 IC50 > 11000 nM T94033 CS2L1Y 21366575 IC50 > 11000 nM T94033 CX1WM9 21366579 IC50 > 11000 nM T94033 CA63IO 21706943 Ki = 450 nM T94033 C80JYP 21707001 Ki = 1300 nM T94033 C5JD2U 21707080 Ki = 5200 nM T94033 CI0SJ2 21967345 Ki = 210 nM T94033 CF4JN6 22010099 Ki > 1000000 nM T94033 C7ZA4U 22010100 Ki > 1000000 nM T94033 CFO41P 22010118 Ki = 123000 nM T94033 C0MI4Y 22038750 Ki = 1600 nM T94033 CAS92P 22038873 Ki = 5500 nM T94033 CJ81IS 22039255 Ki = 74 nM T94033 C7VD8G 22039455 Ki = 85 nM T94033 CD2I7L 22039678 Ki = 7300 nM T94033 C5K6SW 22086973 Ki = 380 nM T94033 CB6IP5 22086976 Ki = 43 nM T94033 CDVH80 22086981 Ki = 130 nM T94033 CLH7A0 22086982 Ki = 58 nM T94033 CG4ZH7 22086988 Ki = 120 nM T94033 CKT23G 22125586 Ki = 1100 nM T94033 CA3I4Y 22280766 Ki = 5200 nM T94033 CSQ96D 22336121 IC50 = 35.39 nM T94033 C7R9CD 22336127 IC50 = 50 nM T94033 C1R9CX 22336133 IC50 = 50 nM T94033 CHOQ30 22336142 IC50 = 42.12 nM T94033 CVG29W 22336143 IC50 = 16.07 nM T94033 CB7N4X 22336146 IC50 = 50 nM T94033 C8URK9 22336148 IC50 = 17.9 nM T94033 C3QEL8 22336150 IC50 = 8.02 nM T94033 C5O7VB 22336151 IC50 = 14.99 nM T94033 C19NAE 22336153 IC50 = 11.82 nM T94033 CHG0A5 22336163 IC50 = 9.4 nM T94033 CTOR48 22336172 IC50 = 50 nM T94033 C51FCG 22336174 IC50 = 70.4 nM T94033 CXZ92L 22336180 IC50 = 19.17 nM T94033 C85UYR 22336181 IC50 = 19.88 nM T94033 CN6P9I 22394409 IC50 = 190 nM T94033 COLY72 22556932 Ki = 43 nM T94033 C2V1NP 22556955 Ki = 25 nM T94033 C4YL7S 22556963 Ki = 40 nM T94033 C9VXC8 22556983 Ki = 260 nM T94033 CA3FT7 22612508 Ki > 5000 nM T94033 CUXK90 22628841 Ki = 10500 nM T94033 CK3GJ4 22665632 IC50 = 28000 nM T94033 C7SJ9B 22665658 IC50 = 48000 nM T94033 CMXF83 22665728 IC50 = 630 nM T94033 CV9D4C 22665887 IC50 = 357000 nM T94033 C4W0GT 22713568 Ki = 10900 nM T94033 CZ58OA 22722451 Ki = 749 nM T94033 CC51MR 22722515 Ki = 86.6 nM T94033 CMDP23 22722517 Ki = 13.2 nM T94033 CREO69 22722585 Ki = 34.6 nM T94033 CJ4W9Q 22722603 Ki = 4.8 nM T94033 CFJ0A9 22722662 Ki = 9.9 nM T94033 CUT8P6 22722666 Ki = 29.7 nM T94033 C2IEN6 22861511 Ki = 1.3 nM T94033 CM2JZ0 22861512 IC50 = 8400 nM T94033 CN3ZI2 22883539 Ki > 4000 nM T94033 CW8EH6 22883547 Ki > 4000 nM T94033 CA3N9L 22883564 Ki = 3100 nM T94033 C9DB7V 22883573 Ki > 4000 nM T94033 CVZ15N 22883583 Ki > 4000 nM T94033 C1R0UD 22883585 Ki > 4000 nM T94033 C13-JAN 22883594 Ki = 1100 nM T94033 CX3IZ5 22946302 Ki = 470 nM T94033 CFH8Y9 22946303 Ki = 171 nM T94033 CIG21R 22985411 Ki = 10 nM T94033 C5Q1GL 22985416 Ki = 15.85 nM T94033 CV13BW 23206211 Ki = 40 nM T94033 CCVI13 23206305 Ki = 6 nM T94033 C3VZ7S 23283289 Ki = 570 nM T94033 CV5NL8 23283331 Ki = 460 nM T94033 C6P9MI 23551902 Ki = 461.9 nM T94033 CPF43A 23586040 Ki = 4100 nM T94033 CQ70HF 23586156 IC50 = 1.39 nM T94033 CNIC40 23629655 Ki = 56100 nM T94033 C7FSW5 23634528 IC50 > 9200 nM T94033 C1JXS8 23634638 Ki = 11000 nM T94033 C0W2EP 23634640 Ki = 100 nM T94033 CD7C1W 23634756 Ki = 4600 nM T94033 C2KJ0P 23634757 Ki = 9400 nM T94033 C6Z9WS 23634758 Ki = 950 nM T94033 C92VIM 23634877 Ki = 4800 nM T94033 CY3NC8 23634878 Ki = 1800 nM T94033 CP6Y7K 23634881 Ki = 12000 nM T94033 C61GCE 23635132 Ki = 980 nM T94033 C75GTN 23635133 Ki = 970 nM T94033 C7HOG9 23635260 Ki = 1000 nM T94033 CR9BK5 23635261 Ki > 6300 nM T94033 CDHQ47 23635262 Ki > 6300 nM T94033 C1KCZ6 23635264 Ki > 6300 nM T94033 CR8AK4 23635386 Ki = 3900 nM T94033 C7U9XO 23635500 Ki = 2520 nM T94033 C8URE5 23635503 Ki = 7000 nM T94033 CH9F4R 23635626 Ki = 12000 nM T94033 CA07TV 23635750 Ki = 1900 nM T94033 CA7Q4T 23635752 Ki > 6300 nM T94033 C06FJI 23635753 Ki > 13400 nM T94033 CTS9W8 23636240 Ki = 180 nM T94033 C50TMW 23636367 Ki = 980 nM T94033 C04CKF 23636368 Ki > 20000 nM T94033 C7JF0K 23636371 Ki = 140 nM T94033 C1XJP6 23644677 Ki = 120 nM T94033 CZ86DS 23644678 Ki = 1.4 nM T94033 C92MUL 23646153 Ki = 800 nM T94033 CJ9OA4 23646154 Ki = 75 nM T94033 CP23GI 23646155 Ki = 97 nM T94033 CH1LX7 23646156 Ki = 57 nM T94033 C83QCW 23646157 Ki = 150 nM T94033 CX8FL0 23646158 Ki = 59 nM T94033 C05YBQ 23646159 Ki = 71 nM T94033 CYB83X 23646160 Ki = 280 nM T94033 CZS9J8 23646161 Ki = 230 nM T94033 C7OC4K 23646163 Ki = 72 nM T94033 CA8EP1 23646164 Ki = 130 nM T94033 CVF49W 23646165 Ki = 250 nM T94033 CGVJ65 23646181 Ki = 330 nM T94033 CN1Q7D 23646208 Ki = 600 nM T94033 CL14AX 23646231 Ki > 63000 nM T94033 C96UDO 23646233 Ki = 13000 nM T94033 C6RM8B 23646234 Ki = 4200 nM T94033 C2U0RB 23646236 Ki = 4200 nM T94033 CPMW70 23646237 Ki > 6300 nM T94033 CS5CV9 23646239 Ki > 270 nM T94033 CV1HY5 23646241 Ki = 390 nM T94033 C6BG3M 23646243 Ki = 4200 nM T94033 CU2V7C 23646245 Ki > 6300 nM T94033 CRX19I 23646295 Ki = 250 nM T94033 CCRD27 23646312 Ki = 130 nM T94033 C1WE6B 23646315 Ki = 130 nM T94033 CDYF29 23646329 IC50 = 2600 nM T94033 CQB29J 23646453 Ki > 35000 nM T94033 C74AMD 23646454 Ki = 2900 nM T94033 CZ7JM9 23646455 Ki = 8600 nM T94033 CD9UH7 23646456 Ki = 9500 nM T94033 CX5S3K 23646457 Ki = 11300 nM T94033 CEH94J 23646458 Ki = 8800 nM T94033 C1DRZ7 23646459 Ki = 4600 nM T94033 CK64IY 23646460 Ki = 10200 nM T94033 CSY57G 23646463 Ki = 1700 nM T94033 C4CV7B 23646580 Ki = 0.12 nM T94033 CJX41O 23646581 Ki = 3.8 nM T94033 C3HT5Y 23646582 Ki = 0.18 nM T94033 C6S4DV 23646583 Ki = 13 nM T94033 CIK6O4 23646584 Ki = 24 nM T94033 C28AXY 23646586 Ki = 0.36 nM T94033 CW4SC7 23646587 Ki = 1.1 nM T94033 C0Z9XE 23646588 Ki = 0.46 nM T94033 CT19DF 23646589 Ki = 73 nM T94033 CNU83K 23646592 IC50 > 100000 nM T94033 CP5Y7A 23646593 Ki = 21 nM T94033 C4TYG1 23646594 Ki = 0.34 nM T94033 COQ28D 23646595 Ki = 380 nM T94033 CJZG27 23646599 Ki = 9.6 nM T94033 C3N9DW 23646600 Ki = 8.1 nM T94033 CPW9D7 23646601 Ki = 6.2 nM T94033 C2HF6N 23646604 Ki = 9.1 nM T94033 CE2ZB5 23646605 Ki = 4.5 nM T94033 CY01NW 23646606 Ki = 3.4 nM T94033 C40RBN 23646607 Ki = 0.58 nM T94033 CU4SI6 23646608 Ki = 0.14 nM T94033 C4R8GB 23646609 Ki = 0.23 nM T94033 CB8ZO2 23646610 Ki = 0.15 nM T94033 C6Q9MH 23646611 Ki = 0.37 nM T94033 C0XO3H 23646612 IC50 = 5 nM T94033 CAIL62 23646615 Ki = 1.5 nM T94033 CSFH79 23646622 Ki = 280 nM T94033 C35HJA 23646623 Ki = 410 nM T94033 C7E4SA 23646732 Ki = 460 nM T94033 C1L9VZ 23647194 IC50 = 620 nM T94033 CC29KT 23647198 IC50 = 370 nM T94033 C9AG8L 23647650 Ki = 1200 nM T94033 CI6N8M 23647676 Ki > 5000 nM T94033 C2QNL5 23647679 Ki = 3200 nM T94033 CEP2K3 23647680 Ki = 1100 nM T94033 CS08RA 23647681 Ki > 5000 nM T94033 CQDG25 23647682 Ki = 2400 nM T94033 CLSE92 23655741 IC50 = 26700 nM T94033 CQ53MU 23655742 IC50 > 9500 nM T94033 C4DOR0 23655937 IC50 > 41300 nM T94033 CRA46X 23655938 IC50 = 21500 nM T94033 CG3W5Q 23661706 IC50 > 30000 nM T94033 CKH4O5 24180463 Ki = 4020 nM T94033 CH5Y8G 24203365 IC50 = 25000 nM T94033 CBXC05 24424330 IC50 = 0.103 nM T94033 CVO5L6 24748791 IC50 = 17000 nM T94033 CUAY58 24749175 IC50 = 390 nM T94033 CL2PU5 24750417 IC50 = 11900 nM T94033 C69OVW 24752832 IC50 = 2600 nM T94033 CI93ZB 24752833 IC50 = 29000 nM T94033 C9DZ3E 24779756 Ki = 0.7 nM T94033 CJSO87 24849206 Ki > 25000 nM T94033 CF7VA8 24858772 Ki = 5.8 nM T94033 C6W5XL 24858773 Ki = 11 nM T94033 CES0Y3 24858774 Ki = 6.5 nM T94033 C9N8CR 24858929 Ki = 3.6 nM T94033 C7QK4H 24858930 Ki = 3.4 nM T94033 CWX43I 24858931 Ki = 2730 nM T94033 CNAG78 24858932 Ki = 2.6 nM T94033 C8RHA3 24858933 Ki = 2940 nM T94033 CQ3S4W 24860438 IC50 > 50000 nM T94033 C5XS4U 24860441 IC50 > 50000 nM T94033 CDWB15 24860442 IC50 > 50000 nM T94033 C4CO3J 24860444 IC50 > 50000 nM T94033 C47AEF 24860445 IC50 > 50000 nM T94033 C9ZS8C 24860446 IC50 > 50000 nM T94033 CNX32B 24860447 IC50 > 50000 nM T94033 CL0W1H 24860448 IC50 > 50000 nM T94033 C0UA9T 24860449 IC50 > 50000 nM T94033 CD8Z9B 24860450 IC50 > 50000 nM T94033 C52CJA 24860451 IC50 > 50000 nM T94033 COX4A7 24873356 Ki = 4700 nM T94033 CC9IQ3 24963037 Ki = 1180 nM T94033 C3BD4T 24997732 Ki > 25000 nM T94033 CN0ZW3 24999867 Ki > 1000 nM T94033 CEM32W 25001205 Ki > 1000 nM T94033 CE6MF2 25022639 Ki = 1.2 nM T94033 CTB92Z 25022661 IC50 = 23 nM T94033 CAO2V4 25030840 Ki = 1400 nM T94033 CU82IO 25030929 Ki = 5100 nM T94033 C7MCT6 25031099 Ki = 71700 nM T94033 C5PO7A 25031100 Ki = 14000 nM T94033 CH7Z1K 25031101 Ki = 670 nM T94033 CEW9X2 25031102 Ki = 600 nM T94033 C9NC4S 25031541 Ki = 270 nM T94033 CK5R8Q 25032200 Ki = 1250 nM T94033 CG8HY2 25032202 Ki = 2100 nM T94033 CH76XK 25032204 Ki = 5100 nM T94033 C07BZQ 25107507 Ki = 9890 nM T94033 CK3FM6 25107508 Ki = 24200 nM T94033 CN3I9J 25107569 Ki = 118000 nM T94033 CB6H7T 25107570 Ki = 320 nM T94033 CC40FO 25107571 Ki = 42 nM T94033 C1QC4Y 25107572 Ki = 220 nM T94033 CKJ04T 25107573 Ki = 670 nM T94033 CN8Y0B 25107634 Ki = 156 nM T94033 C84XCZ 25107635 Ki = 190 nM T94033 CCY26A 25107636 Ki = 490 nM T94033 CO03GM 25107637 Ki = 4930 nM T94033 CNR43C 25107638 Ki = 5000 nM T94033 CDAC04 25107705 Ki = 5160 nM T94033 CYS45L 25107706 Ki = 3980 nM T94033 CYS98D 25107707 Ki = 1760 nM T94033 CRV78W 25107708 Ki = 740 nM T94033 CF85WU 25107709 Ki = 60 nM T94033 C23YAU 25107770 Ki = 25 nM T94033 CQZ70E 25107771 Ki = 2860 nM T94033 CEK7G5 25107772 Ki = 16900 nM T94033 C3V7JU 25107773 Ki = 620 nM T94033 CBYN26 25107774 Ki = 5500 nM T94033 CI90TE 25113126 Ki = 6810 nM T94033 CVL17T 25113128 Ki = 180 nM T94033 C0ZRB1 25113615 Ki = 750 nM T94033 CUVH16 25113616 Ki = 5000 nM T94033 C7NT1J 25113617 Ki = 1000 nM T94033 CWE9U5 25134248 Ki = 1170 nM T94033 CAEM12 25147483 Ki = 14000 nM T94033 C2H4PJ 25166809 Ki > 13000 nM T94033 CG76TR 25181493 Ki = 40 nM T94033 CKM7Y8 25269170 Ki > 20000 nM T94033 CY4FG8 36596148 Ki = 581000 nM T94033 CU5YR1 41583852 IC50 > 200000 nM T94033 CQ76OP 42615253 Ki = 109000 nM T94033 CKA8D5 42615254 Ki = 100 nM T94033 CVAI06 42643068 Ki = 2800 nM T94033 CUF74S 42643069 Ki = 8600 nM T94033 CZ03OW 42643070 Ki > 35000 nM T94033 CZ7M8C 42643120 Ki = 5900 nM T94033 C0KN2D 42643121 Ki = 15300 nM T94033 CL6GN4 42643122 Ki > 35000 nM T94033 C54UVP 43165100 Ki = 2511886.43 nM T94033 CA81RS 44144381 Ki = 0.29 nM T94033 C8ZJ0B 44156919 IC50 = 370 nM T94033 CPX15D 44188281 IC50 = 39.7 nM T94033 CR8W6M 44200855 IC50 = 28 nM T94033 C4TZ2X 44201094 IC50 = 12 nM T94033 CZ2V5J 44237081 Ki = 180 nM T94033 CAOU89 44237086 Ki = 100 nM T94033 C3J2IC 44249750 IC50 = 0.084 ug.mL-1 T94033 CGQ24J 44263948 Ki = 1500 nM T94033 C7PLD3 44264049 Ki > 20000 nM T94033 C9OMR4 44264598 Ki = 19 nM T94033 CD5QB6 44264609 Ki = 4500 nM T94033 CI0J6S 44264612 Ki = 2200 nM T94033 CZV98I 44264619 Ki = 49000 nM T94033 CT5PS4 44264627 Ki = 300 nM T94033 C5V9OZ 44264631 Ki = 3400 nM T94033 C25ZLT 44264637 Ki = 1500 nM T94033 CW39RT 44264643 Ki = 31 nM T94033 CRK37Z 44264650 Ki = 220 nM T94033 C9RND0 44264660 Ki = 27 nM T94033 C9M4WX 44264663 Ki = 84 nM T94033 CW7ZH4 44264664 Ki = 105 nM T94033 CPI2K3 44264665 Ki = 4 nM T94033 C9TA6F 44264681 Ki = 1.8 nM T94033 C9D6UJ 44264685 Ki > 20000 nM T94033 CAVJ67 44264698 Ki = 32 nM T94033 C03CAW 44264699 Ki = 12 nM T94033 CPRE58 44264710 Ki = 0.53 nM T94033 CA8N9H 44264719 Ki = 0.05 nM T94033 C6OZ8E 44264778 Ki = 5.8 nM T94033 C6SH1P 44264790 IC50 = 340 nM T94033 CPFD24 44264795 Ki = 47 nM T94033 CW1G8N 44264814 Ki = 0.02 nM T94033 CF49JR 44264817 Ki = 2.2 nM T94033 C6IDX1 44264832 Ki = 0.5 nM T94033 CT40BD 44264834 Ki = 5.3 nM T94033 CKGY06 44264842 Ki = 6 nM T94033 C1YVD9 44264854 Ki = 2.4 nM T94033 C3NTZ1 44264856 IC50 = 1060 nM T94033 C2XLN7 44264885 Ki = 19000 nM T94033 CW4R8J 44264888 Ki = 6200 nM T94033 CT2V6S 44264889 Ki = 17000 nM T94033 CZDW40 44264920 Ki = 6600 nM T94033 C9RZ0O 44264921 Ki = 18000 nM T94033 CXQ1H9 44264935 Ki > 21000 nM T94033 C6O5VF 44264936 Ki = 800 nM T94033 CVBG38 44264940 Ki > 21000 nM T94033 C63WPN 44264954 Ki > 21000 nM T94033 CB3AQ1 44264955 Ki > 6300 nM T94033 CGCI69 44264981 Ki > 21000 nM T94033 C78WPK 44264995 Ki > 6300 nM T94033 C01WIT 44265005 Ki = 14000 nM T94033 C1BP7E 44265006 Ki > 21000 nM T94033 CQNX29 44265034 Ki = 5900 nM T94033 C4YZ2K 44265893 Ki = 0.3 nM T94033 CJBG39 44265902 Ki = 0.38 nM T94033 C4DS8K 44265936 Ki = 3.3 nM T94033 C24GFJ 44265937 Ki = 0.045 nM T94033 CW85TJ 44265948 Ki = 3.8 nM T94033 CY8H6F 44265957 Ki = 3300 nM T94033 C95DZG 44265958 Ki = 11 nM T94033 C2RGV9 44265960 Ki = 8 nM T94033 CY1M7B 44265961 Ki = 0.12 nM T94033 C3EF4P 44265996 Ki = 18.4 nM T94033 CPU8Q6 44266026 Ki = 0.1 nM T94033 C6OJ4I 44266844 Ki = 0.21 nM T94033 CB4ZN6 44266860 Ki = 0.084 nM T94033 C4LWN5 44266873 Ki = 0.4 nM T94033 COA64J 44268334 Ki = 1540 nM T94033 C3Y1IS 44268338 Ki = 575 nM T94033 CO84YQ 44268339 Ki = 12 nM T94033 CZB60J 44268342 Ki = 81 nM T94033 CPG17Z 44268343 Ki = 36 nM T94033 C3CTV2 44268344 Ki = 26 nM T94033 CLPK74 44268345 Ki = 43 nM T94033 C3HYX1 44268356 Ki = 1610 nM T94033 CP0KF4 44268360 Ki = 280 nM T94033 CKH94X 44268361 Ki = 82 nM T94033 CZ67LH 44268362 Ki = 41 nM T94033 CZ2D9V 44268392 Ki = 100 nM T94033 C9I2UE 44268393 Ki = 16 nM T94033 CYQH61 44268411 Ki = 69 nM T94033 CP0RZ5 44268414 Ki = 6510 nM T94033 CAK75M 44268426 Ki = 11930 nM T94033 CIX56V 44268441 Ki = 11810 nM T94033 C5G6UO 44269720 Ki = 14000 nM T94033 CGX38A 44271471 IC50 = 970 nM T94033 C6H5KB 44271477 IC50 = 6000 nM T94033 CIBJ02 44271491 IC50 = 240 nM T94033 CTV0Y1 44271544 IC50 = 4900 nM T94033 CA4OP3 44272421 Ki = 276.2 nM T94033 CRMS45 44272522 Ki = 196.8 nM T94033 C6NP4Y 44272594 Ki = 3.2 nM T94033 C3HOE9 44272634 Ki = 1.1 nM T94033 C16LZF 44272637 Ki = 5.5 nM T94033 C8D3CM 44272663 Ki = 5.9 nM T94033 C9CYW3 44272664 Ki = 9.8 nM T94033 C5TP2L 44272674 Ki = 140.8 nM T94033 CKZ6O0 44272690 Ki = 136 nM T94033 CA61IM 44272691 Ki = 323.8 nM T94033 CT9XH1 44272744 Ki = 20.8 nM T94033 C3S5BW 44272813 Ki = 13.2 nM T94033 CB64EA 44272825 Ki = 0.1 nM T94033 C7QGZ3 44272858 Ki = 103.2 nM T94033 CJ2L7A 44272860 Ki = 357.1 nM T94033 CQ3LX2 44272873 Ki = 30.8 nM T94033 CP32GC 44273614 IC50 = 4800 nM T94033 C8C1WF 44273817 IC50 = 590 nM T94033 CCJN68 44273818 IC50 = 260 nM T94033 CR3V4S 44273853 IC50 = 1400 nM T94033 CN4HE5 44273854 IC50 = 48 nM T94033 C90AKQ 44273901 IC50 = 19400 nM T94033 CL7NY5 44274017 IC50 = 5500 nM T94033 C7I2DQ 44274065 IC50 = 3100 nM T94033 CMG90C 44274089 IC50 > 10000 nM T94033 CPZ6X4 44274830 Ki = 5 nM T94033 C2NI3X 44274840 Ki = 1995 nM T94033 CO7Z3E 44274843 Ki = 5000 nM T94033 C7FP2X 44274865 Ki = 5000 nM T94033 CNZ83L 44274886 Ki = 2000 nM T94033 C9UP2G 44274929 Ki = 610 nM T94033 C9WDV8 44274930 Ki > 5000 nM T94033 C3U8OC 44274931 Ki = 870 nM T94033 C2U5SO 44274945 Ki = 5000 nM T94033 CVJ28M 44274963 Ki = 631 nM T94033 CK0RZ3 44274987 Ki = 4 nM T94033 C0XIV9 44275030 Ki = 158 nM T94033 CQ0TN7 44275052 Ki = 316 nM T94033 CPE28K 44275084 Ki = 50 nM T94033 C5VE6G 44275194 Ki > 5000 nM T94033 CT2J0P 44275195 Ki > 5000 nM T94033 C42RVS 44275227 Ki = 2600 nM T94033 CQ12EP 44275238 Ki = 2500 nM T94033 C3OM8S 44275239 Ki = 75 nM T94033 CGOH67 44275240 Ki = 380 nM T94033 CU52WR 44275243 Ki = 3500 nM T94033 C2HO4D 44275249 Ki = 200 nM T94033 C1N5GM 44275254 Ki = 1120 nM T94033 CX1C4Q 44275257 Ki = 1960 nM T94033 C9EKZ2 44275271 Ki = 880 nM T94033 C4TBU7 44275275 Ki > 5000 nM T94033 C2D9YK 44275287 Ki = 770 nM T94033 CPBU68 44275289 Ki = 22 nM T94033 CL4D3K 44275297 Ki > 5000 nM T94033 C3LS5P 44275326 Ki = 1500 nM T94033 CHJC81 44275330 Ki = 190 nM T94033 C4SO5M 44275345 Ki = 3600 nM T94033 CBA9T0 44275361 Ki = 210 nM T94033 CEWU09 44275365 Ki > 5000 nM T94033 CHP2T5 44276502 IC50 = 2000 nM T94033 C3HP6D 44276503 IC50 = 2400 nM T94033 CBL97R 44276508 IC50 = 59000 nM T94033 C3MDB2 44276519 IC50 = 66000 nM T94033 CL30JE 44276604 IC50 = 15000 nM T94033 C4ZG2R 44276629 IC50 = 36000 nM T94033 CNB07T 44276630 IC50 = 19000 nM T94033 C7CK0J 44276899 IC50 = 92.1 nM T94033 C9TD3J 44277049 Ki = 0.16 nM T94033 C9U5MT 44277050 Ki = 0.85 nM T94033 CFOL73 44277057 Ki = 0.087 nM T94033 CD5F2Q 44277058 Ki = 3.6 nM T94033 CVU1T9 44277085 IC50 = 284 nM T94033 CHV5J6 44277135 Ki = 2.5 nM T94033 C79EHD 44277167 Ki = 7 nM T94033 CS8IO2 44277200 Ki = 1.7 nM T94033 CH73LJ 44277220 Ki = 0.19 nM T94033 CMFG14 44277228 Ki = 1.1 nM T94033 CY98IU 44277248 Ki = 1.3 nM T94033 CVK7H4 44277254 Ki = 2 nM T94033 C46CSH 44277277 Ki = 3 nM T94033 C62TUQ 44277332 IC50 > 2500 nM T94033 C6FW1R 44277353 Ki = 3 nM T94033 CCZ16D 44277358 Ki = 3.6 nM T94033 CML2Q1 44277359 Ki = 4.8 nM T94033 CJ6NH1 44277373 Ki = 5.2 nM T94033 CHZ2Q4 44277564 IC50 > 2500 nM T94033 C19OGX 44278104 IC50 = 1.2 nM T94033 C7UZI2 44278318 Ki = 0.31 nM T94033 C1MTC4 44278351 Ki = 0.073 nM T94033 C2CU6D 44278352 Ki = 0.071 nM T94033 C9OW3M 44278353 Ki = 2000 nM T94033 C6U7YV 44278433 Ki = 0.45 nM T94033 CCTX01 44281308 Ki = 28 nM T94033 CAY28E 44281309 Ki = 13 nM T94033 CN38WH 44281319 Ki = 0.75 nM T94033 CJ1U4H 44281323 Ki = 0.27 nM T94033 CA41LW 44281326 Ki = 0.24 nM T94033 CQG5S1 44281327 Ki = 24 nM T94033 C7VRF5 44281335 Ki = 4.7 nM T94033 C9L0RF 44281355 Ki = 0.32 nM T94033 CZ6B9G 44281376 Ki = 30 nM T94033 C9Z5NY 44281377 Ki = 87 nM T94033 CD46SY 44281388 Ki = 0.087 nM T94033 CED25A 44281394 Ki = 5.7 nM T94033 CZ93CF 44281401 Ki = 32 nM T94033 C6ZJH7 44281406 Ki = 83 nM T94033 CZX9E5 44281421 Ki = 82 nM T94033 CKO48Z 44281490 Ki = 11 nM T94033 CLW39A 44281506 Ki = 29 nM T94033 C0GKV7 44281518 Ki = 18 nM T94033 C4JSO7 44281550 Ki = 78 nM T94033 CLD9W4 44281552 Ki = 53 nM T94033 C2AE4O 44281566 Ki = 80 nM T94033 C3H9CA 44281580 Ki = 1.2 nM T94033 CIUM69 44281581 Ki = 3.8 nM T94033 CAJB43 44281595 Ki = 1.7 nM T94033 C5HG3X 44281617 Ki = 7.7 nM T94033 CBY79Z 44281618 Ki = 39 nM T94033 C1L9TK 44281622 Ki = 91 nM T94033 CWCL75 44281623 Ki = 1.5 nM T94033 C0WC2D 44281640 Ki = 53 nM T94033 CY4OH1 44281648 Ki = 32 nM T94033 C0T7OQ 44281652 Ki = 94 nM T94033 CLBK42 44281661 Ki = 0.057 nM T94033 C07WBX 44281669 Ki = 15 nM T94033 C5B9UC 44281675 Ki = 36 nM T94033 CRD83W 44281707 Ki = 2.9 nM T94033 CP21EY 44281709 Ki = 1.5 nM T94033 C9LK8J 44281725 Ki = 17 nM T94033 C07TZM 44281805 Ki = 3 nM T94033 C9QJD3 44281806 Ki = 28 nM T94033 C4M5RL 44281807 Ki = 22 nM T94033 CFY4G7 44282088 Ki = 0.023 nM T94033 C4A1ZJ 44282153 Ki > 100000 nM T94033 C5DZ4L 44282601 Ki = 11200 nM T94033 CRT93X 44282678 Ki > 50000 nM T94033 CA6X2L 44283195 Ki > 50000 nM T94033 CSIQ87 44283615 IC50 = 5440 nM T94033 CHN6X0 44283616 IC50 = 190 nM T94033 CML1T6 44283635 IC50 = 9 nM T94033 CM90WC 44283786 Ki = 5 nM T94033 C2JMY1 44283808 Ki = 47 nM T94033 C6DFY9 44283892 Ki = 49.3 nM T94033 C73PDT 44283894 Ki = 39.4 nM T94033 CE0NG1 44283905 Ki = 4.6 nM T94033 C7QU0Y 44283909 Ki = 77 nM T94033 CPM23R 44283911 Ki = 403 nM T94033 CMFT95 44283921 Ki = 47 nM T94033 CLGI45 44283936 Ki = 29 nM T94033 CAJX21 44283999 Ki = 166 nM T94033 C0QSL6 44284108 Ki = 114 nM T94033 CVR6P4 44284109 Ki = 137 nM T94033 C3WPL2 44284147 Ki = 95 nM T94033 CF49EI 44284150 Ki = 102 nM T94033 C2NRA3 44284163 Ki = 690 nM T94033 C5IEZ1 44284242 Ki = 31 nM T94033 CK87LW 44284376 Ki = 32.4 nM T94033 CR6QO5 44284377 Ki = 364 nM T94033 CMU9A4 44284541 IC50 = 650 nM T94033 CXK3M6 44284559 IC50 = 2200 nM T94033 C36PXQ 44284752 IC50 = 1600 nM T94033 C8Y9JZ 44284991 Ki = 0.028 nM T94033 CMZ71H 44284992 Ki = 0.019 nM T94033 CV2I0Y 44285015 Ki = 29 nM T94033 CAY3Z9 44285016 Ki = 7 nM T94033 C6USR4 44285077 Ki = 20 nM T94033 C5NU9L 44285118 Ki = 0.027 nM T94033 CG0F6A 44285119 Ki = 11000 nM T94033 C4GM5N 44285174 Ki = 43 nM T94033 CU9G2F 44285211 Ki = 0.007 nM T94033 C0FPN1 44285253 Ki = 0.002 nM T94033 C9N1ZL 44285281 Ki = 0.011 nM T94033 CV15DH 44285283 Ki = 1000 nM T94033 CMKJ72 44285284 Ki = 21 nM T94033 CYTC82 44285311 Ki = 19 nM T94033 C5PX3O 44285312 Ki = 0.059 nM T94033 C7ZRS5 44285351 Ki = 25 nM T94033 C9LRW8 44285352 Ki = 0.082 nM T94033 C2OSN4 44285775 Ki = 310 nM T94033 CWBZ82 44286069 Ki = 30 nM T94033 C2TKY1 44286104 Ki = 130 nM T94033 C92POZ 44286346 Ki = 77 nM T94033 CGC79Q 44286347 Ki = 94 nM T94033 C8CDV0 44286348 Ki = 82 nM T94033 C1V9UA 44286349 Ki = 500 nM T94033 CLAO70 44286351 Ki = 39 nM T94033 CEUX40 44286370 Ki = 125 nM T94033 CEM0X2 44286371 Ki = 34 nM T94033 CMOW21 44286372 Ki = 34 nM T94033 C5N0YB 44286374 Ki = 27 nM T94033 C79GIH 44286375 Ki = 119 nM T94033 C4R5BH 44286398 Ki = 64 nM T94033 CQ82ZW 44286426 IC50 = 141 nM T94033 COPR02 44286428 IC50 = 2.32 nM T94033 CS5U7F 44286453 IC50 = 0.467 nM T94033 CPJ52V 44286627 Ki = 47 nM T94033 CSCT34 44286628 Ki = 47300 nM T94033 C8OSI3 44286658 Ki = 3100 nM T94033 C5S2RT 44286683 Ki = 359 nM T94033 CD83AF 44286684 Ki = 723 nM T94033 CPK5M6 44286709 Ki = 32 nM T94033 CQ2AD1 44286777 Ki = 4560 nM T94033 C2IUQ3 44286788 Ki = 6700 nM T94033 C4HY3W 44286804 Ki = 780 nM T94033 CK84NJ 44286805 Ki = 452 nM T94033 C7GL2H 44286832 Ki = 1570 nM T94033 CC9G2D 44286852 Ki = 26 nM T94033 CQ2A3R 44286878 Ki = 95 nM T94033 CJP7K9 44286879 Ki = 430 nM T94033 CHZM39 44286931 Ki = 2190 nM T94033 C6M7BW 44286944 Ki = 760 nM T94033 C6YHF8 44286960 Ki = 810 nM T94033 CRK53N 44286978 Ki = 85 nM T94033 C7WU5K 44287028 Ki = 150 nM T94033 CMA2Q6 44287039 Ki = 1600 nM T94033 C0DG5R 44287043 Ki = 248 nM T94033 CGPL91 44287130 Ki = 59900 nM T94033 C5Q0TP 44287162 Ki = 3280 nM T94033 C63JTG 44287260 IC50 > 500000 nM T94033 CB9D2R 44287527 IC50 > 100000 nM T94033 CCXM09 44287610 IC50 > 100000 nM T94033 CB8IQ5 44287628 IC50 = 39000 nM T94033 CT4N0L 44287629 IC50 = 64000 nM T94033 C0G3DY 44287647 Ki = 0.92 nM T94033 C9IC3S 44287667 Ki = 0.46 nM T94033 CQ75ND 44287668 Ki = 0.36 nM T94033 CS5D4G 44287745 IC50 = 50000 nM T94033 CL5I1S 44287757 IC50 = 42000 nM T94033 CXEC79 44287771 IC50 = 106 nM T94033 C3QD4W 44287797 Ki = 260 nM T94033 C5W7SA 44287798 Ki = 320 nM T94033 CX47AK 44287838 IC50 > 500000 nM T94033 C5Q9OJ 44287854 IC50 = 200 nM T94033 C5UT7J 44287855 IC50 = 2000 nM T94033 CDTY78 44287882 Ki = 0.21 nM T94033 COI15D 44287916 Ki = 10 nM T94033 C6QP1H 44287919 Ki = 512 nM T94033 C02ARM 44287937 Ki = 33 nM T94033 CN59QG 44287940 Ki = 6.9 nM T94033 C2N6JE 44287941 Ki = 110 nM T94033 CMY2L6 44287943 Ki = 42 nM T94033 CPD6J7 44287944 Ki = 30 nM T94033 CO95FJ 44287962 Ki = 8.3 nM T94033 CJH70N 44287992 Ki = 3.5 nM T94033 C9B3EF 44287995 Ki = 26 nM T94033 C4NJE9 44287996 Ki = 19 nM T94033 C7UQ9V 44287997 Ki = 1.1 nM T94033 CP90NM 44288029 Ki = 1.3 nM T94033 C73CRM 44288039 Ki = 410 nM T94033 CUHK16 44288040 Ki = 580 nM T94033 CA02GU 44288104 Ki = 0.94 nM T94033 C0P8SV 44288201 Ki = 2000 nM T94033 C8AEQ2 44288202 Ki = 9900 nM T94033 CV8BX7 44288203 Ki = 170000 nM T94033 C4UQZ8 44288223 Ki = 5.5 nM T94033 C1NUA2 44288243 Ki = 1.3 nM T94033 CF9X4J 44288274 Ki = 1.2 nM T94033 CIG0D7 44288309 Ki = 0.42 nM T94033 C2V4LF 44288413 Ki = 137 nM T94033 C2XO1U 44288435 Ki = 1.7 nM T94033 C3AUV9 44288524 IC50 = 48000 nM T94033 C9XAR3 44288526 Ki = 1.7 nM T94033 CB02UK 44288572 IC50 = 20200 nM T94033 CI6JM8 44288931 Ki = 630 nM T94033 C02WNS 44288932 Ki = 6400 nM T94033 C10IJH 44288953 Ki = 7000 nM T94033 CPA63F 44288982 Ki = 6500 nM T94033 C7JH5R 44288983 Ki = 9000 nM T94033 CQ7BY9 44289132 Ki = 423000 nM T94033 CWR03N 44289153 Ki = 386000 nM T94033 CBU7X1 44289180 Ki = 561000 nM T94033 C0YV7U 44289263 Ki > 1000000 nM T94033 C1Q7KW 44289264 Ki > 1000000 nM T94033 CD1TP0 44289295 Ki = 94400 nM T94033 C75NCO 44289296 Ki = 52900 nM T94033 CWZL84 44289297 Ki > 1000000 nM T94033 CUQ35M 44289336 Ki = 41200 nM T94033 CONY81 44289354 Ki = 31900 nM T94033 C49UIC 44289570 Ki = 340 nM T94033 CQ8KM3 44289599 Ki = 2100 nM T94033 CC0S4X 44289600 Ki = 15 nM T94033 CI0G4E 44289615 Ki = 7 nM T94033 CMS2Z1 44289616 Ki = 7.4 nM T94033 CYZ76X 44289617 Ki = 8.5 nM T94033 C18PCW 44289618 Ki = 0.07 nM T94033 C7Q6YH 44289619 Ki = 900 nM T94033 C97TBS 44289631 Ki = 12 nM T94033 C1H8GD 44289632 Ki = 18 nM T94033 CZRH12 44290033 IC50 > 11000 nM T94033 CUY95P 44290108 IC50 > 11000 nM T94033 CS76AC 44290361 IC50 = 380 nM T94033 CMY82L 44290376 IC50 = 11000 nM T94033 CHL9Y6 44290377 IC50 = 3000 nM T94033 CLDH85 44290378 IC50 = 660 nM T94033 CXO05N 44290379 IC50 = 43000 nM T94033 CNWI90 44290501 IC50 > 200000 nM T94033 CBE24K 44290502 IC50 = 13000 nM T94033 C94BSK 44290516 IC50 = 3200 nM T94033 CAXB95 44290518 IC50 = 5000 nM T94033 C49EPA 44290519 IC50 = 50 nM T94033 C37IJH 44290520 IC50 = 130 nM T94033 C30GAZ 44290521 IC50 = 4000 nM T94033 CU17NH 44290529 IC50 = 5600 nM T94033 CC8YQ3 44290530 IC50 = 16 nM T94033 CN04WY 44290542 IC50 = 12000 nM T94033 CF8JK0 44290543 Ki = 709 nM T94033 C05EYJ 44290555 IC50 = 16 nM T94033 C10ANS 44290556 IC50 = 5000 nM T94033 CO9JQ0 44290557 Ki > 4000 nM T94033 CY60EW 44290560 Ki > 4000 nM T94033 C70XKC 44290569 Ki > 4000 nM T94033 CEO13F 44290576 IC50 = 49000 nM T94033 C9QS3I 44290584 Ki > 4000 nM T94033 CUW14A 44290648 Ki = 650 nM T94033 COB93L 44290673 Ki > 4000 nM T94033 C2UV6T 44290696 Ki > 3950 nM T94033 C8LY1J 44290712 Ki > 3950 nM T94033 C0SYK2 44290731 Ki = 990 nM T94033 CN6KP1 44290929 Ki > 4000 nM T94033 C0E1RV 44290930 Ki = 2660 nM T94033 C8APX2 44290947 Ki > 4000 nM T94033 CXWY26 44290963 Ki = 0.49 nM T94033 CZ7PT1 44290965 Ki > 4000 nM T94033 CTA7I1 44291034 Ki = 4000 nM T94033 CH59WK 44291046 Ki = 2800 nM T94033 CYFC04 44291049 Ki > 4000 nM T94033 C7TNE0 44291050 Ki > 4000 nM T94033 CC4RN5 44291077 Ki > 4000 nM T94033 CXKG43 44291143 Ki = 91 nM T94033 C9XAE5 44291144 Ki = 60 nM T94033 CV3Q8F 44291293 Ki = 1.25 nM T94033 C9RBW1 44291445 Ki = 0.84 nM T94033 CU5QR7 44291783 Ki = 185 nM T94033 CGU75L 44291826 Ki = 310 nM T94033 C2IK7H 44291827 Ki = 21 nM T94033 CX9I6H 44291828 Ki = 0.19 nM T94033 CA9TP1 44292003 Ki = 160 nM T94033 C67GIO 44292022 Ki = 58 nM T94033 CMO16W 44292151 Ki > 500000 nM T94033 C7DT0R 44292384 Ki > 10000 nM T94033 C2JQ3O 44292951 Ki = 16 nM T94033 CW02PO 44292952 Ki = 12 nM T94033 CL5VP0 44293219 Ki = 0.12 nM T94033 C60GBH 44293221 Ki = 2.6 nM T94033 CE0QR2 44293262 Ki = 4 nM T94033 CC26FY 44293263 Ki = 26 nM T94033 CXV2U0 44293745 Ki > 5000 nM T94033 CYHM09 44293746 Ki > 5000 nM T94033 CWZ6Y0 44294144 Ki > 5000 nM T94033 C5AZX1 44294161 Ki > 5000 nM T94033 C5P8QF 44294202 Ki = 1200 nM T94033 C0O2PG 44295723 Ki = 750 nM T94033 C6U9CB 44295788 Ki = 12000 nM T94033 C7SN2O 44295812 Ki = 2500 nM T94033 C8AY9O 44296035 Ki = 6600 nM T94033 CLK7N1 44296052 Ki = 78000 nM T94033 CQ51FN 44296074 Ki = 6900 nM T94033 CETN87 44296078 Ki = 700000 nM T94033 C3DG0L 44296128 Ki = 330 nM T94033 CPF86Z 44296129 Ki = 710 nM T94033 C38SDX 44296130 Ki = 23000 nM T94033 C1WU8B 44296135 Ki = 440 nM T94033 CV31AF 44296181 Ki > 5000 nM T94033 C6Y2TQ 44296217 Ki = 336 nM T94033 C9UG6P 44296249 Ki = 320 nM T94033 C2IPC9 44296275 Ki = 16 nM T94033 C83JPT 44296276 Ki = 18 nM T94033 CUF3Y8 44296306 Ki = 13 nM T94033 C5YLG9 44296316 Ki = 63 nM T94033 CH58EX 44296342 Ki = 12 nM T94033 CHEY58 44296365 Ki = 48 nM T94033 CXL8T3 44296383 Ki = 80 nM T94033 CDHG78 44296386 Ki = 15 nM T94033 C1BM0O 44296439 Ki = 300 nM T94033 C9HM6D 44296481 Ki = 43 nM T94033 C2RVU1 44296502 Ki = 11 nM T94033 CTE04W 44296503 Ki = 10 nM T94033 C9AGW7 44297775 Ki = 1000000 nM T94033 C5HX1A 44297783 Ki = 800000 nM T94033 C9R1GP 44301401 Ki > 10000 nM T94033 CFJT06 44301437 Ki = 83 nM T94033 CD48UC 44301440 Ki > 10000 nM T94033 CD52XY 44301522 Ki > 10000 nM T94033 CH39US 44301758 IC50 = 70000 nM T94033 C29MVU 44303719 Ki > 450000 nM T94033 C3FB4I 44303721 Ki = 315000 nM T94033 CQLA16 44303733 Ki > 450000 nM T94033 C5RZL0 44303743 Ki = 7500 nM T94033 CTE75P 44303769 Ki = 34000 nM T94033 C16GOI 44303778 Ki = 9500 nM T94033 C26ZUK 44303789 Ki = 12000 nM T94033 CN6V9A 44303803 Ki = 10000 nM T94033 C67ZRW 44303804 Ki = 120000 nM T94033 CB38WA 44303805 Ki = 23000 nM T94033 CL0U1A 44303806 Ki = 8000 nM T94033 CVO2D9 44303808 Ki = 185000 nM T94033 C0JZY5 44303810 Ki = 29000 nM T94033 CFJ4W3 44303811 Ki = 14000 nM T94033 CE0R9A 44303824 Ki > 450000 nM T94033 C5YF7O 44303839 Ki > 450000 nM T94033 C2LY4T 44303843 Ki = 1000 nM T94033 C3HXW6 44303858 Ki = 320 nM T94033 CYW9S8 44303912 Ki > 450000 nM T94033 CIQZ37 44303925 Ki > 450000 nM T94033 CJN72A 44303933 Ki = 9000 nM T94033 CXCY31 44303935 Ki = 195000 nM T94033 C4SN8T 44304006 Ki > 450000 nM T94033 CL16JC 44304046 Ki > 450000 nM T94033 CAM6R0 44304047 Ki > 450000 nM T94033 CR4V0L 44304084 Ki = 310000 nM T94033 CG37DH 44304086 Ki = 330000 nM T94033 C7UJH1 44304087 Ki = 43000 nM T94033 CG0R8N 44304097 Ki = 205000 nM T94033 CJ80KE 44304098 Ki > 450000 nM T94033 CG8TI6 44304099 Ki > 450000 nM T94033 C9W8QC 44304100 Ki > 450000 nM T94033 CE31BF 44304104 Ki > 450000 nM T94033 C9XIO1 44304105 Ki > 450000 nM T94033 C83YIU 44304139 Ki = 125000 nM T94033 CP5S9K 44304192 Ki = 450000 nM T94033 CKD98A 44304353 Ki > 450000 nM T94033 C09HMY 44305854 IC50 = 3.2 nM T94033 C9OQ6V 44305961 IC50 > 10 nM T94033 C6DSU1 44307502 IC50 > 530000 nM T94033 C5A7KQ 44307505 IC50 = 17600 nM T94033 CIOB75 44307762 IC50 = 30000 nM T94033 CDNM94 44308631 IC50 = 2300 nM T94033 C2FYA6 44308649 IC50 = 24000 nM T94033 CPYN65 44308650 IC50 = 470 nM T94033 CBQX97 44308779 IC50 = 2500 nM T94033 CW84QO 44310082 IC50 = 4600 nM T94033 C5VER7 44310204 IC50 = 1400 nM T94033 CTOD17 44310306 IC50 = 110 nM T94033 CMG13A 44310471 IC50 = 4300 nM T94033 CS0ZI8 44310936 IC50 = 7.2 nM T94033 CI36UV 44310952 IC50 = 10 nM T94033 CH0G4Y 44310953 IC50 = 31.7 nM T94033 CS0WU6 44310956 IC50 = 8600 nM T94033 C5W7JY 44311005 IC50 = 4600 nM T94033 CDIJ45 44311021 IC50 = 13 nM T94033 CN7SV6 44311065 IC50 = 1350 nM T94033 CKV48X 44311294 IC50 = 24 nM T94033 C54MRA 44311312 IC50 = 4.9 nM T94033 C86SDO 44311314 IC50 = 21.6 nM T94033 C6L2FG 44311333 IC50 = 14 nM T94033 CZ87WQ 44311437 IC50 = 3 nM T94033 CKP5W7 44311564 IC50 > 1100 nM T94033 C6TQ7D 44312627 IC50 > 10000 nM T94033 CTW03S 44312639 IC50 = 4090 nM T94033 C18PFJ 44312776 IC50 > 10000 nM T94033 CGS74O 44312851 IC50 > 10000 nM T94033 CM5RQ6 44312966 IC50 > 10000 nM T94033 CGND24 44312967 IC50 > 10000 nM T94033 CRN7I3 44313020 IC50 > 10000 nM T94033 C3X7VO 44313132 IC50 = 6 nM T94033 C6G0NQ 44313284 IC50 > 10000 nM T94033 CYQ4I0 44313285 IC50 > 10000 nM T94033 C2D0JU 44313317 IC50 > 10000 nM T94033 CR12HS 44313338 IC50 = 10 nM T94033 CM6L5C 44313347 IC50 = 10 nM T94033 C8T0BL 44313350 IC50 = 3800 nM T94033 C9OQN5 44313404 IC50 = 92 nM T94033 CU8S5P 44313405 IC50 = 6 nM T94033 CHU84X 44313413 IC50 = 66 nM T94033 CIQ1L7 44313498 IC50 = 18 nM T94033 CF1S3C 44313499 IC50 = 16 nM T94033 C0G3WT 44313500 IC50 = 600 nM T94033 C1KQR4 44313688 Ki = 3600 nM T94033 C87HJP 44313722 IC50 = 12 nM T94033 C3H5RB 44313873 IC50 > 2500 nM T94033 C8V3IH 44313932 IC50 > 2500 nM T94033 C6VP5I 44314000 IC50 > 2500 nM T94033 CT2ZD9 44314001 IC50 = 2210 nM T94033 CFXW28 44314002 IC50 = 1960 nM T94033 CM10DN 44314053 IC50 > 2500 nM T94033 CCK1W8 44314117 IC50 = 1720 nM T94033 CT1X8J 44314118 IC50 = 3830 nM T94033 C5H6VU 44314181 IC50 > 2500 nM T94033 CSTP54 44314265 IC50 > 2500 nM T94033 CN8WP6 44314436 Ki = 0.035 nM T94033 CP20SA 44314437 Ki = 1.58 nM T94033 C3IBT0 44314446 Ki = 1.89 nM T94033 CX78CW 44314654 Ki = 5.09 nM T94033 C21QLG 44314683 Ki = 18 nM T94033 C0U2WD 44314684 Ki = 0.3 nM T94033 CY3V0H 44314874 Ki = 0.2 nM T94033 C9IN4E 44314967 IC50 = 110 nM T94033 C0Z8UC 44315048 Ki = 4.33 nM T94033 C4Q9ZF 44315391 Ki > 1000000 nM T94033 C87MBQ 44315392 Ki = 274000 nM T94033 C5CIL6 44315449 Ki = 363000 nM T94033 C2QOP6 44315450 Ki = 34000 nM T94033 C5WI0G 44315604 Ki > 1000000 nM T94033 CDW83E 44315605 Ki > 1000000 nM T94033 CIBE78 44315607 Ki > 1000000 nM T94033 CZ3CY0 44315608 Ki > 1000000 nM T94033 C07NBY 44315609 Ki > 1000000 nM T94033 C8DQ5R 44315610 Ki > 1000000 nM T94033 C0Z7PI 44315635 Ki > 1000000 nM T94033 CJ5I9T 44315636 Ki > 1000000 nM T94033 C71UBD 44315637 Ki > 1000000 nM T94033 C8UAJ1 44315641 Ki > 1000000 nM T94033 CH7M1F 44315642 Ki > 1000000 nM T94033 C0EG4V 44315643 Ki > 1000000 nM T94033 C8MU4G 44315644 Ki > 1000000 nM T94033 C2U5HM 44315664 Ki = 138000 nM T94033 CPT78A 44315674 Ki > 1000000 nM T94033 CEO18C 44315675 Ki > 1000000 nM T94033 C25DGE 44315677 Ki > 1000000 nM T94033 C45PHT 44315678 Ki > 1000000 nM T94033 C5QUO9 44315743 Ki = 492000 nM T94033 CA8L4R 44315744 Ki > 1000000 nM T94033 CPV7S5 44315758 Ki > 1000000 nM T94033 CRVN48 44315788 Ki = 269000 nM T94033 C1QEV6 44315805 Ki > 1000000 nM T94033 CB7Q2W 44315826 Ki > 1000000 nM T94033 CPH5U7 44315831 Ki > 1000000 nM T94033 CG3VB1 44315832 Ki > 1000000 nM T94033 CZ8RS4 44315843 Ki > 1000000 nM T94033 CUGF09 44315844 Ki > 1000000 nM T94033 CX20QR 44315845 Ki = 14000 nM T94033 C4KF3H 44315846 Ki > 1000000 nM T94033 CCXE57 44315848 Ki > 1000000 nM T94033 C0IVD5 44315849 Ki > 1000000 nM T94033 CU74AZ 44315850 Ki > 1000000 nM T94033 C9QO7H 44315851 Ki > 1000000 nM T94033 CF4I7B 44315852 Ki > 1000000 nM T94033 CS6C5I 44315912 Ki = 741000 nM T94033 CF48NZ 44315913 Ki > 1000000 nM T94033 C6O5ZT 44315914 Ki > 1000000 nM T94033 C8VZ4J 44315915 Ki > 1000000 nM T94033 CZ6K5W 44316015 Ki > 1000000 nM T94033 CUL40O 44316026 Ki > 1000000 nM T94033 CAJ97K 44316048 Ki > 1000000 nM T94033 CQ52SH 44316049 Ki > 1000000 nM T94033 C1MRI0 44316050 Ki > 1000000 nM T94033 CV38TK 44316051 Ki > 1000000 nM T94033 CKWY45 44316065 Ki > 1000000 nM T94033 CKN8C1 44316486 IC50 = 430 nM T94033 C97NYB 44317783 IC50 = 1375 nM T94033 C5AK3D 44317785 IC50 = 31.9 nM T94033 CK5XV4 44318022 Ki = 2280 nM T94033 CFCJ83 44318038 IC50 = 193 nM T94033 CW2X9Z 44318052 IC50 = 466 nM T94033 C90NPX 44318079 Ki = 130 nM T94033 CBQ0D2 44318098 Ki = 55 nM T94033 C57VSJ 44318156 IC50 = 160 nM T94033 CK58VB 44318182 IC50 = 1.1 nM T94033 CV8IB4 44318218 IC50 = 130 nM T94033 C1C0UG 44318220 IC50 = 1800 nM T94033 CK5RC4 44318223 IC50 = 2.07 nM T94033 COV05F 44318305 Ki = 140 nM T94033 CP2QJ5 44318465 Ki = 200 nM T94033 C7C8BZ 44319291 Ki ~ 4000 nM T94033 C2X7AE 44319684 Ki = 60.5 nM T94033 C62CXR 44319685 Ki = 5.7 nM T94033 C6D3SA 44319701 Ki = 20.1 nM T94033 C4P6WI 44319919 Ki = 9.6 nM T94033 CMS05A 44319941 Ki = 107 nM T94033 CM4XP3 44320181 Ki = 10.1 nM T94033 CEZ84L 44320397 IC50 > 2500 nM T94033 CD5IN8 44320423 Ki = 3.1 nM T94033 CSK62O 44320493 IC50 = 192 nM T94033 CYT2Q4 44320495 IC50 > 2500 nM T94033 CG36WH 44320752 IC50 = 285 nM T94033 CQ64CD 44320839 IC50 = 235 nM T94033 CK1EZ2 44320862 IC50 = 178 nM T94033 C7AMH4 44320876 IC50 = 0.71 nM T94033 C8XF3O 44322227 Ki = 1 nM T94033 CX73RG 44324726 Ki = 9300 nM T94033 CMZ05T 44324727 Ki > 21000 nM T94033 CI5BY6 44324744 Ki > 21000 nM T94033 CKDN47 44324745 Ki > 21000 nM T94033 CWN4P7 44325526 Ki > 4000 nM T94033 C1MT8R 44325527 Ki > 4000 nM T94033 CBD24R 44325803 Ki = 0.045 nM T94033 CZW79L 44325865 Ki > 4000 nM T94033 C4Q8AC 44325938 Ki > 4000 nM T94033 C61VAC 44325939 Ki > 4000 nM T94033 CK92AD 44325940 Ki > 4000 nM T94033 C5TLH0 44325953 Ki > 4000 nM T94033 CHI47Q 44325959 Ki = 1200 nM T94033 C1DES8 44325967 Ki > 4000 nM T94033 C5CLJ1 44325971 Ki = 1400 nM T94033 CYOQ97 44325982 Ki > 4000 nM T94033 C3A2IO 44325983 Ki > 4000 nM T94033 CO2F4Z 44326181 Ki > 4000 nM T94033 CF92WZ 44326243 Ki = 3900 nM T94033 C90VZO 44326339 Ki = 6100 nM T94033 CZU3E4 44326592 Ki = 0.31 nM T94033 C4JVD5 44326631 Ki = 3 nM T94033 CA24BR 44326766 Ki = 0.74 nM T94033 CJ05KH 44326777 Ki = 2.6 nM T94033 CC73LK 44326853 Ki = 44 nM T94033 C2V7CW 44326854 Ki = 208 nM T94033 CCB8G9 44326877 Ki = 480 nM T94033 CVX1M4 44326890 Ki = 29 nM T94033 CC1FI5 44326899 Ki = 24 nM T94033 CUEY50 44326920 Ki = 12 nM T94033 CQ34BR 44326924 Ki = 15 nM T94033 CJT7H6 44326928 Ki > 20000 nM T94033 CS1HG3 44326938 Ki > 20000 nM T94033 C0I4SV 44326961 Ki = 0.8 nM T94033 CAG6M5 44327046 Ki = 1.3 nM T94033 C3NIJ1 44327069 Ki = 5 nM T94033 CFV5D6 44327462 Ki = 2200 nM T94033 CI56QW 44327465 Ki = 11100 nM T94033 CTDM97 44327484 Ki = 11200 nM T94033 C86YFO 44327490 Ki = 2200 nM T94033 CE3UL6 44327872 Ki = 11800 nM T94033 C5Q8SZ 44328328 IC50 = 1400 nM T94033 CWR3M9 44328445 IC50 = 560 nM T94033 CY7G8N 44328503 IC50 = 209000 nM T94033 C51DLA 44328525 IC50 = 5000 nM T94033 CBO8W3 44328590 IC50 = 6000 nM T94033 CRPE62 44328622 IC50 = 1580 nM T94033 C8C4YO 44330249 Ki = 80 nM T94033 C3K4OG 44330356 Ki = 5 nM T94033 CTKP16 44330409 IC50 = 90000 nM T94033 C26KJP 44330423 Ki = 4.9 nM T94033 CVR6K0 44330453 IC50 = 20 nM T94033 C5W1DZ 44330605 IC50 = 170 nM T94033 C76ZOE 44330607 IC50 = 7200 nM T94033 C6B0DP 44330620 IC50 = 210 nM T94033 CN70HF 44330627 Ki = 4.68 nM T94033 CW1XE9 44330628 Ki = 1.4 nM T94033 C1Z5FA 44330631 Ki = 0.16 nM T94033 CK8FJ6 44330632 Ki = 9.1 nM T94033 CT2K9N 44330633 Ki = 123 nM T94033 CS1V3W 44330665 Ki = 1.71 nM T94033 CQX7A3 44330666 Ki = 2.1 nM T94033 C4LC7K 44330667 Ki = 0.8 nM T94033 CJC2P7 44330822 Ki = 5.4 nM T94033 CYT0C9 44330823 Ki = 16 nM T94033 CWV7X5 44330835 Ki = 0.69 nM T94033 C98KLH 44330847 Ki = 1.6 nM T94033 CSM3B6 44330879 IC50 > 10000 nM T94033 CVM21A 44330906 IC50 > 10000 nM T94033 CY72JW 44330907 IC50 > 10000 nM T94033 CA4Y1P 44330934 IC50 > 10000 nM T94033 CTSB26 44330953 Ki = 159 nM T94033 C9XC5H 44330954 Ki = 15 nM T94033 C3K6JA 44330969 IC50 = 880 nM T94033 CXW57P 44330970 IC50 = 1000 nM T94033 CU9Z4M 44330999 IC50 = 3200 nM T94033 C9KW3Q 44331002 IC50 > 10000 nM T94033 CJ9Y8Z 44331003 IC50 > 10000 nM T94033 C1X4UM 44331004 IC50 > 10000 nM T94033 C2SK9N 44331021 IC50 = 6000 nM T94033 C2CS3N 44331022 IC50 = 1300 nM T94033 CAB5T7 44331052 IC50 = 820 nM T94033 CVM80P 44331070 Ki = 20 nM T94033 CR7F8L 44331114 IC50 > 10000 nM T94033 C4NP5G 44331140 IC50 > 10000 nM T94033 CSDQ73 44331145 IC50 > 10000 nM T94033 C4CJ5M 44331146 IC50 > 10000 nM T94033 CFK17Y 44331147 IC50 > 10000 nM T94033 C5SDZ6 44331170 Ki = 9.9 nM T94033 CQ4S2Z 44331171 Ki = 86 nM T94033 CO27PQ 44331172 Ki = 163 nM T94033 C2BS5N 44331180 IC50 > 10000 nM T94033 C90GYM 44331181 Ki = 3.1 nM T94033 CE7TD9 44331182 Ki = 5.3 nM T94033 C1NR3B 44331189 IC50 = 10000 nM T94033 CF13OL 44331190 IC50 > 10000 nM T94033 CE69GW 44331194 IC50 > 10000 nM T94033 C3SU1R 44331210 IC50 > 10000 nM T94033 CM63UN 44331224 Ki = 473 nM T94033 C6O7JE 44331225 Ki = 1800 nM T94033 C6L2OQ 44331247 Ki = 24 nM T94033 C0YOA6 44331389 IC50 = 21 nM T94033 CGL57V 44331419 IC50 = 16800 nM T94033 C6OPK8 44331423 IC50 > 100000 nM T94033 CTB69R 44331436 IC50 = 19 nM T94033 C4E9VP 44332474 Ki = 30 nM T94033 C35EKA 44332921 Ki = 1.06 nM T94033 CJAL34 44332934 Ki = 1.8 nM T94033 CZF4G0 44332981 Ki = 2 nM T94033 CSJ82M 44333044 Ki = 0.4 nM T94033 CN1P5Y 44333061 Ki = 0.33 nM T94033 CC48QN 44333068 Ki = 14 nM T94033 C79CIZ 44333147 EC50 = 1170 nM T94033 CQHE08 44333168 EC50 = 390 nM T94033 CQ35OB 44333225 EC50 = 590 nM T94033 CMQ72Z 44333240 EC50 = 590 nM T94033 CDI42N 44333242 EC50 = 56000 nM T94033 CHRI62 44333246 EC50 = 150 nM T94033 CLTW49 44333255 EC50 = 880 nM T94033 CNGD56 44333258 EC50 = 49 nM T94033 CC3RU7 44333259 EC50 = 840 nM T94033 C2K5HZ 44333803 Ki = 16000 nM T94033 C5M2LB 44333833 Ki > 50000 nM T94033 CYNL31 44333951 Ki = 1.2 nM T94033 C0FE1Y 44333960 Ki = 2.4 nM T94033 CJ2IM6 44333972 Ki = 0.89 nM T94033 CNF52U 44333992 Ki = 0.43 nM T94033 CIO79X 44334002 Ki = 0.36 nM T94033 CTUX56 44334003 Ki = 0.42 nM T94033 CS5X8Z 44334242 Ki = 0.06 nM T94033 CYX2N3 44334264 Ki = 0.06 nM T94033 CNTU54 44334314 Ki = 0.3 nM T94033 CDMP53 44334315 Ki = 0.58 nM T94033 CI3CT4 44334316 Ki = 0.53 nM T94033 CL05HM 44334318 Ki = 3 nM T94033 CN4TX8 44334349 Ki = 0.83 nM T94033 CQA75Y 44334374 Ki = 0.28 nM T94033 CI0C4V 44334382 Ki = 0.41 nM T94033 C7Y8IG 44334488 Ki = 610 nM T94033 C0O1XG 44334554 Ki = 0.37 nM T94033 CHL01I 44334805 Ki = 1100 nM T94033 CAI31R 44334928 IC50 = 55 nM T94033 C1A2EL 44334931 IC50 = 19 nM T94033 C8BKP0 44335014 IC50 = 25 nM T94033 CJFL84 44335118 IC50 = 27 nM T94033 CI43YO 44336084 Ki = 1460 nM T94033 C4HJR3 44336093 Ki = 280 nM T94033 CS1TA7 44336150 Ki = 159 nM T94033 CHQE05 44336151 Ki = 135 nM T94033 CT8H9V 44336606 Ki = 500 nM T94033 CM2C9Q 44336608 Ki = 900 nM T94033 C5V6AE 44336618 Ki = 600 nM T94033 CE83LV 44336620 Ki = 300 nM T94033 C6PO3F 44336653 Ki = 900 nM T94033 CRQB16 44336655 Ki = 1800 nM T94033 CWGK84 44336668 Ki = 300 nM T94033 CP5BG3 44336674 Ki = 15000 nM T94033 C5Y9NM 44336676 Ki = 9000 nM T94033 COPT26 44336682 Ki = 1400 nM T94033 CLE10Q 44336690 Ki = 17000 nM T94033 C9LI2J 44336719 Ki = 6100 nM T94033 C7M9PA 44336735 Ki = 3500 nM T94033 CHM49Q 44337735 Ki = 2500 nM T94033 CV7HW5 44337751 Ki = 120 nM T94033 CDS43Z 44337779 Ki = 34000 nM T94033 C39GBZ 44337785 Ki = 11800 nM T94033 CX35DM 44337794 Ki = 6900 nM T94033 CN1WI2 44337821 Ki = 25000 nM T94033 CE27KP 44337862 IC50 = 260 nM T94033 C61CGV 44337884 IC50 = 18 nM T94033 C4EFA8 44337894 IC50 = 55 nM T94033 C0HP3T 44337899 IC50 = 78000 nM T94033 CH0K1J 44337917 IC50 = 27 nM T94033 CG6T9S 44337925 IC50 = 5100 nM T94033 CA10BE 44337935 IC50 = 3600 nM T94033 C4ATV2 44337945 IC50 = 23 nM T94033 C2AN5G 44337986 IC50 = 28 nM T94033 CFH80Q 44337989 IC50 = 250 nM T94033 CTD5Q8 44338012 IC50 = 130 nM T94033 C5OVP7 44338032 IC50 = 94 nM T94033 CGD65V 44338048 IC50 = 72 nM T94033 CI8U6O 44338109 IC50 = 2.3 nM T94033 C9WR3T 44338140 IC50 = 3200 nM T94033 CSUB92 44338144 Ki = 50 nM T94033 CZW8I0 44338156 IC50 > 2500 nM T94033 C9P8UK 44338157 IC50 = 13200 nM T94033 C7KM8P 44338170 IC50 = 22100 nM T94033 C4ZKD5 44338177 Ki = 18 nM T94033 CNI7P4 44338191 Ki = 3 nM T94033 CY29AD 44338192 Ki = 0.35 nM T94033 CUD4G3 44338355 IC50 > 2500 nM T94033 C04MBF 44338376 IC50 = 880 nM T94033 CRMU28 44338377 IC50 > 2500 nM T94033 CA1G6Q 44338381 IC50 = 12800 nM T94033 CN6SV4 44338385 Ki = 0.5 nM T94033 C1KEZ2 44338386 Ki = 0.5 nM T94033 CW6R1A 44338455 Ki = 0.106 nM T94033 CW25JV 44338459 Ki = 16 nM T94033 CI70HX 44338476 Ki = 3 nM T94033 C5O0HW 44338486 Ki = 58 nM T94033 C6C3NY 44338487 Ki = 0.5 nM T94033 C52BLN 44338495 Ki = 2.5 nM T94033 C4F9LY 44338503 Ki = 0.5 nM T94033 CMJ45D 44338511 Ki = 4.4 nM T94033 C27IMO 44338512 Ki = 3 nM T94033 CQ6P3H 44338513 Ki = 0.96 nM T94033 CL61JK 44338564 Ki = 25 nM T94033 CEF91D 44338589 Ki = 32 nM T94033 C05AVM 44338604 Ki = 16 nM T94033 CUJ32E 44338605 Ki = 5 nM T94033 C5K8UW 44338606 Ki = 24 nM T94033 C8BTX2 44338607 Ki = 1.2 nM T94033 CA42TW 44338624 Ki = 0.92 nM T94033 CFXN40 44338644 Ki = 17 nM T94033 CHX17O 44339365 Ki = 2300 nM T94033 CSA5H1 44339376 Ki = 1340 nM T94033 CZR56N 44339399 Ki = 157 nM T94033 C4AZH1 44339401 Ki = 3800 nM T94033 C9B0SQ 44339404 Ki = 102 nM T94033 CC2K4G 44339417 Ki = 100 nM T94033 C5WZ9O 44339442 Ki = 77 nM T94033 C0G3LP 44339443 Ki = 652 nM T94033 C4CZ2V 44339453 Ki = 42 nM T94033 C7E4KL 44339464 Ki = 1440 nM T94033 CV53DA 44339470 Ki = 22 nM T94033 CAY91C 44339490 Ki = 19 nM T94033 CB6R0I 44339610 Ki = 1160 nM T94033 C7TOG2 44339650 Ki = 562 nM T94033 CU04CH 44339859 Ki = 5300 nM T94033 C6GB0R 44339860 Ki = 51000 nM T94033 CH8KX0 44340005 Ki = 88000 nM T94033 CRL13W 44340006 Ki = 32000 nM T94033 C5KD1P 44340079 Ki = 24000 nM T94033 COE58R 44340086 Ki = 230000 nM T94033 C9O8MH 44340114 Ki = 82000 nM T94033 C5FC2M 44340115 Ki = 28000 nM T94033 CGL01I 44340240 Ki = 22000 nM T94033 C7WU5B 44340241 Ki = 29000 nM T94033 CFO32G 44340290 Ki = 85000 nM T94033 CF50ZE 44340291 Ki = 23000 nM T94033 CO1B2F 44340292 Ki = 32000 nM T94033 C6G7CA 44341184 Ki = 3.5 nM T94033 CKA1T3 44341287 IC50 = 1.1 nM T94033 CZ9BF5 44341288 IC50 = 16.4 nM T94033 C4XEK1 44341417 IC50 = 5.01 nM T94033 C72DOW 44341724 Ki = 1300 nM T94033 CXL2Q8 44341827 Ki = 200 nM T94033 C1I9EN 44342050 Ki = 1700 nM T94033 CTH60L 44342051 Ki = 11600 nM T94033 CQ2PR0 44342242 Ki > 100000 nM T94033 C2AT7J 44342409 Ki = 1400 nM T94033 CNW1B2 44342560 IC50 = 1 nM T94033 C2Z7SD 44342561 IC50 = 150 nM T94033 CM7G1U 44342634 IC50 = 77 nM T94033 CQW48S 44342644 IC50 = 137 nM T94033 CCYN38 44342736 IC50 = 33 nM T94033 C26UXG 44342977 IC50 = 10715.19 nM T94033 CC0Z8V 44343581 IC50 > 2500 nM T94033 CW76HT 44343582 IC50 = 2500 nM T94033 CD0TW8 44343615 IC50 > 2500 nM T94033 C9NZE1 44343799 IC50 > 2500 nM T94033 CAIZ35 44343800 IC50 > 2500 nM T94033 C0W6EI 44343845 IC50 > 2500 nM T94033 C46IGW 44343852 IC50 > 2500 nM T94033 C5H3NY 44343853 IC50 > 2500 nM T94033 C7B5GK 44343857 IC50 > 2500 nM T94033 C40EHX 44343858 IC50 = 1270 nM T94033 C91PVF 44343859 IC50 = 1770 nM T94033 C4MS5Q 44343972 IC50 > 2500 nM T94033 C3ZI7A 44343993 IC50 = 2500 nM T94033 CMEI89 44343994 IC50 > 2500 nM T94033 CEA17Z 44344039 IC50 > 2500 nM T94033 CUO74X 44344054 IC50 > 2500 nM T94033 CIG0Q2 44344067 Ki = 130 nM T94033 CQ7R5F 44344069 Ki = 49 nM T94033 CANQ97 44344083 Ki = 5.2 nM T94033 C52JVD 44344096 Ki = 313 nM T94033 CBTF46 44344097 Ki = 4.1 nM T94033 C60GZW 44344100 IC50 = 537 nM T94033 CAJT87 44344125 Ki = 3.3 nM T94033 C93EWF 44344138 Ki = 490 nM T94033 C0B1CU 44344151 Ki = 3.3 nM T94033 C6CDJ3 44344152 Ki = 6.6 nM T94033 CREZ48 44344153 IC50 > 2500 nM T94033 CRYS42 44344167 Ki = 470 nM T94033 CK9YA3 44344184 Ki = 0.13 nM T94033 C1LS3Q 44344185 Ki = 62 nM T94033 CJH5K8 44345610 Ki = 19 nM T94033 CO4C6L 44345611 Ki = 72 nM T94033 C74WFZ 44345628 Ki = 25 nM T94033 CM2YO1 44345652 Ki > 4000 nM T94033 C76GKC 44345708 Ki = 48 nM T94033 CTG52Z 44345709 Ki = 45 nM T94033 CI6JS9 44345710 Ki = 43 nM T94033 CFET03 44345727 Ki = 19 nM T94033 CZ0KR4 44345728 Ki = 19 nM T94033 CIG6D9 44345740 Ki = 49 nM T94033 CZD14B 44345741 Ki = 110 nM T94033 CY2UM3 44345923 Ki = 27 nM T94033 CV5NA9 44345928 Ki = 634 nM T94033 C3TFS9 44345929 Ki = 33 nM T94033 CJ5ZL0 44345930 Ki = 18 nM T94033 CD7Y2K 44345955 Ki = 15 nM T94033 CPT06F 44345968 IC50 = 240 nM T94033 CF10WJ 44345991 Ki = 41 nM T94033 C9KDO7 44345992 Ki = 24 nM T94033 C5I2BL 44345993 Ki = 90 nM T94033 C5D4VP 44346013 Ki = 65 nM T94033 CK05QD 44346026 Ki = 47 nM T94033 CM6U3P 44346044 Ki = 99 nM T94033 C6FLW3 44346045 Ki = 24 nM T94033 CCE5L7 44346049 IC50 = 6000 nM T94033 C87UKY 44346051 IC50 = 10000 nM T94033 C70GNE 44346059 Ki = 49 nM T94033 C5NK1H 44346060 Ki = 35 nM T94033 C1WD0Y 44346061 Ki = 18 nM T94033 C98UPV 44346069 IC50 = 100000 nM T94033 C3NYJ9 44346077 IC50 = 240 nM T94033 C6Q7OK 44346081 IC50 = 100000 nM T94033 C6U2FO 44346150 IC50 = 74000 nM T94033 C60WMZ 44346155 IC50 = 73000 nM T94033 COZ32R 44346156 IC50 = 1100 nM T94033 CLQ1Y2 44346161 IC50 = 100000 nM T94033 CP2E1D 44346163 IC50 = 110 nM T94033 CS5P2K 44346164 IC50 = 13500 nM T94033 C36WLU 44346165 IC50 = 133000 nM T94033 CS63FQ 44346373 Ki = 0.4 nM T94033 C3RBW8 44347347 Ki = 4 nM T94033 CAY34C 44347478 Ki = 3.4 nM T94033 CT0QN1 44347480 Ki = 2.2 nM T94033 C1UN9I 44347534 Ki = 1.8 nM T94033 C0V2FL 44347624 Ki = 0.28 nM T94033 CML27I 44347734 Ki = 147 nM T94033 C6K3ZR 44347735 Ki = 33 nM T94033 CN3VT6 44347748 Ki = 17 nM T94033 C1TUJ6 44347819 Ki = 10 nM T94033 CTQ93K 44347853 Ki = 1600 nM T94033 CA7C9J 44347854 Ki = 400 nM T94033 CT5F1U 44347863 Ki = 28 nM T94033 CDMG63 44347916 Ki = 14500 nM T94033 C7NB1I 44347920 Ki = 204 nM T94033 CEP6C1 44347929 Ki = 12100 nM T94033 CFN61M 44347930 Ki = 156 nM T94033 CAH89Z 44347942 Ki = 68 nM T94033 CCJ1K0 44347943 Ki = 7 nM T94033 CCK84E 44347944 Ki = 8 nM T94033 CC50UP 44347950 Ki = 1900 nM T94033 C0PR3S 44347951 Ki = 14800 nM T94033 C7FUH8 44347960 Ki = 373 nM T94033 CW2B1L 44347973 Ki = 3200 nM T94033 C47TSD 44347978 Ki = 38 nM T94033 CNLT06 44347994 Ki = 23 nM T94033 CK4VR8 44347995 Ki = 16 nM T94033 C7F6BG 44347997 Ki = 4000 nM T94033 CM5P9C 44347998 Ki = 17 nM T94033 CH3BL8 44348002 Ki = 59 nM T94033 CDAJ75 44348003 Ki = 159 nM T94033 CKBN18 44348006 Ki = 2300 nM T94033 CX85LK 44348013 Ki = 6760 nM T94033 CQTB91 44348014 Ki = 3180 nM T94033 CHE69P 44348015 Ki = 65 nM T94033 CXN6O9 44348021 Ki = 9100 nM T94033 C64JUL 44348030 Ki = 11900 nM T94033 CCKQ91 44348032 Ki = 9 nM T94033 CJF76L 44348040 Ki = 8 nM T94033 CKU5T7 44348041 Ki = 6 nM T94033 CC89VP 44348059 Ki = 31 nM T94033 C58MFB 44348077 IC50 > 10000 nM T94033 CJ1XO7 44348087 Ki = 7900 nM T94033 CNI3R5 44348088 Ki = 21 nM T94033 C25GOA 44348089 Ki = 52 nM T94033 CQ8CK5 44348093 Ki > 21000 nM T94033 C5XCE4 44348104 Ki = 195 nM T94033 C2R1PU 44348105 Ki = 24 nM T94033 C31JWA 44348108 Ki = 1600 nM T94033 CWE9T4 44348110 Ki = 6 nM T94033 CPV7C4 44348111 Ki = 500 nM T94033 CDZF52 44348115 Ki = 4 nM T94033 C6QBK5 44348118 Ki = 4 nM T94033 C0I9LG 44348119 Ki = 86 nM T94033 C1X8ZN 44348120 Ki = 73 nM T94033 C73NHB 44348129 Ki = 110 nM T94033 CUM75D 44348141 Ki = 94 nM T94033 C0OQ6V 44348142 Ki = 21 nM T94033 CO5Y7S 44348145 Ki = 650 nM T94033 C1X6WN 44348165 Ki = 22 nM T94033 C6O8NQ 44348177 Ki > 50000 nM T94033 C38CNV 44348180 Ki = 34 nM T94033 C7KID6 44348201 Ki = 20 nM T94033 C9NI3P 44348211 Ki = 52 nM T94033 C8ZCJ2 44348212 Ki = 47 nM T94033 CWV07K 44348217 Ki = 38 nM T94033 CQM0O4 44348226 Ki = 2300 nM T94033 CPD32J 44348228 Ki = 9800 nM T94033 C2ZH8C 44348233 Ki = 213 nM T94033 CH9SP6 44348260 Ki = 91 nM T94033 CH61QP 44348436 IC50 > 10000 nM T94033 CA74EQ 44348505 IC50 > 10000 nM T94033 C2M6TU 44348587 IC50 > 10000 nM T94033 CED0Q4 44348616 IC50 > 10000 nM T94033 CZI93S 44348618 IC50 > 10000 nM T94033 CR68KY 44348619 IC50 > 10000 nM T94033 C5H7ZW 44348620 IC50 > 10000 nM T94033 C94NSH 44348621 IC50 > 10000 nM T94033 CYS5G0 44348624 IC50 > 10000 nM T94033 CFWR38 44348631 IC50 > 10000 nM T94033 CV5F9W 44348635 IC50 > 10000 nM T94033 C6QXM9 44348648 IC50 > 10000 nM T94033 C04CQG 44348722 IC50 > 10000 nM T94033 CBR0V8 44348733 IC50 > 10000 nM T94033 CP2H0Q 44348745 IC50 > 10000 nM T94033 C6T5EP 44349954 Ki = 100 nM T94033 CW20MI 44349969 IC50 = 29 nM T94033 C4G2UO 44350259 Ki = 100 nM T94033 C6BCO4 44350260 Ki = 100 nM T94033 CD8AL2 44351097 IC50 > 200000 nM T94033 CHGE39 44351104 IC50 = 44580 nM T94033 C2RMW4 44351162 IC50 > 100000 nM T94033 CPB5X3 44351901 Ki = 6 nM T94033 CJ2RK7 44351999 Ki = 4.7 nM T94033 CKT1P5 44352000 Ki = 36 nM T94033 CAR0P9 44352005 Ki = 1300 nM T94033 C1GC7N 44352010 Ki = 40 nM T94033 C07XGO 44352011 Ki > 1000 nM T94033 C9XWN4 44352021 Ki = 420 nM T94033 C9C5RY 44352022 Ki = 44 nM T94033 CB0ZP5 44352023 Ki = 9.2 nM T94033 CWZS23 44352024 Ki = 4.4 nM T94033 C1H5DQ 44352025 Ki = 11 nM T94033 C2OH3W 44352031 Ki = 11 nM T94033 C4ZQ8V 44352041 Ki = 20 nM T94033 C2HPA5 44352111 IC50 = 486 nM T94033 CFOA49 44352112 IC50 = 247 nM T94033 CAQ0J4 44352177 IC50 > 32000 nM T94033 CU05JC 44352204 IC50 = 4880 nM T94033 C2A5ZL 44352219 IC50 = 19800 nM T94033 CC0D1E 44352249 IC50 = 164 nM T94033 C5DZV0 44352273 IC50 = 8140 nM T94033 C2F6KR 44352286 IC50 = 130 nM T94033 C4KQH7 44352287 IC50 = 961 nM T94033 CJ18VQ 44353163 IC50 > 30000 nM T94033 C2ET4H 44353164 IC50 = 3210 nM T94033 CD8JT3 44353192 IC50 < 40 nM T94033 CE1RS4 44353237 Ki = 75 nM T94033 C65CXD 44353259 Ki = 3 nM T94033 C6FE1Z 44353295 IC50 > 30000 nM T94033 CM3JI6 44353296 IC50 > 30000 nM T94033 CX9MJ6 44356715 Ki = 14840 nM T94033 CZBU73 44357452 IC50 = 1800 nM T94033 CCA2H8 44357456 IC50 = 1600 nM T94033 C6H9JK 44357484 IC50 = 600 nM T94033 C2QML5 44357515 IC50 = 9 nM T94033 C9RQN6 44357516 IC50 = 77 nM T94033 C45DNJ 44358162 IC50 = 620 nM T94033 C3J0UR 44358222 IC50 = 2800 nM T94033 CA58DF 44358245 IC50 = 1400 nM T94033 C7CB6L 44358272 IC50 = 27000 nM T94033 C52HNW 44358305 IC50 = 110 nM T94033 C47XMA 44358313 IC50 = 500 nM T94033 C1OZ5J 44358321 IC50 = 7400 nM T94033 CWE3U6 44358340 IC50 = 12 nM T94033 CI67FJ 44358341 IC50 = 650 nM T94033 CCI10U 44358363 IC50 = 14000 nM T94033 C8O4BZ 44358364 IC50 = 50 nM T94033 C3F2VU 44358365 IC50 = 80 nM T94033 CLM4G8 44358384 IC50 = 2900 nM T94033 C94NDL 44358386 IC50 = 32 nM T94033 CPY90E 44358398 IC50 = 75 nM T94033 CFP49Z 44358401 IC50 = 200 nM T94033 CQR9B8 44358429 IC50 = 310 nM T94033 C8BC3Z 44358436 Ki = 12500 nM T94033 CPO39C 44358576 Ki = 1500 nM T94033 C2QOY4 44358663 Ki = 0.27 nM T94033 CG89JF 44358782 IC50 = 6200 nM T94033 CHS4B0 44358903 Ki = 28 nM T94033 CVHL15 44359057 IC50 > 100000 nM T94033 C2CH7M 44359059 IC50 = 24200 nM T94033 CG0MW7 44359453 IC50 = 3500 nM T94033 C1KL4Q 44359454 IC50 = 2700 nM T94033 CPU61I 44359598 IC50 = 1700 nM T94033 C2Q1NY 44359626 IC50 = 3800 nM T94033 C82XKL 44359703 IC50 = 1460 nM T94033 CS8AH1 44359715 IC50 = 2500 nM T94033 C29ANK 44359723 Ki = 1.01 nM T94033 CQ5F0T 44359724 IC50 = 709 nM T94033 C4Y5HK 44359726 IC50 = 420 nM T94033 CIKY14 44359730 Ki 0.54 nM T94033 C40POZ 44359735 IC50 = 1.1 nM T94033 CF0V6J 44359754 IC50 = 111 nM T94033 C5P3UG 44359755 IC50 = 157 nM T94033 C5UKJ2 44359756 IC50 = 125 nM T94033 CQ10VZ 44359794 IC50 = 286 nM T94033 C5ES1X 44359805 IC50 = 235 nM T94033 C5CTA0 44359810 Ki 0.85 nM T94033 CSV16F 44359885 IC50 = 0.7 nM T94033 CD3R9Q 44359906 IC50 = 14.2 nM T94033 CERC69 44359907 IC50 > 2500 nM T94033 CMDB96 44360123 IC50 = 159 nM T94033 C9FPE5 44360927 Ki = 66 nM T94033 C2WYS3 44361130 Ki = 280 nM T94033 C52ABN 44361131 Ki = 11 nM T94033 C3AE9R 44363282 IC50 = 8900 nM T94033 C1CM6S 44363283 IC50 = 5200 nM T94033 C8ZYG4 44363379 IC50 = 3000 nM T94033 CVF7J8 44363380 IC50 = 2900 nM T94033 C34FDQ 44363400 IC50 = 4900 nM T94033 C9BNX3 44363401 IC50 = 12000 nM T94033 C8R1BJ 44363428 IC50 = 1400 nM T94033 C6OKF9 44363431 IC50 = 2900 nM T94033 C9SH7B 44363439 IC50 = 3500 nM T94033 C5Q1TB 44363463 IC50 = 26600 nM T94033 C4MGZ1 44363497 IC50 = 108000 nM T94033 CQ4O9C 44363514 IC50 = 110000 nM T94033 C0J6LI 44363534 IC50 > 333000 nM T94033 CI4D5E 44363537 IC50 = 42000 nM T94033 CEU61M 44363592 IC50 = 10 nM T94033 CA46US 44363644 IC50 = 70 nM T94033 C2YME9 44363739 IC50 = 4400 nM T94033 CY07UH 44363753 IC50 = 134000 nM T94033 C2P6RJ 44364043 Ki > 100000 nM T94033 C06RPS 44364101 Ki > 100000 nM T94033 C8H3IU 44364106 Ki > 100000 nM T94033 C0B3TG 44364107 Ki > 100000 nM T94033 CN46VL 44364123 Ki > 100000 nM T94033 C1P0MS 44364177 Ki > 100000 nM T94033 CYK89L 44364205 Ki > 100000 nM T94033 C6VP2F 44364263 Ki = 620 nM T94033 CP7K4W 44364302 Ki > 100000 nM T94033 C4LH6Q 44364310 Ki = 4000 nM T94033 CB85LE 44364311 Ki > 100000 nM T94033 CDE32K 44364319 Ki = 15000 nM T94033 CTC3O5 44364320 Ki = 16000 nM T94033 CSI3V9 44364329 Ki > 100000 nM T94033 CUM70S 44364371 Ki = 8000 nM T94033 C9Z7JD 44364382 Ki > 100000 nM T94033 CT8QM1 44364445 Ki = 20000 nM T94033 CTB86G 44364486 Ki > 100000 nM T94033 C1ELX6 44364487 Ki > 100000 nM T94033 CQ1LM8 44364504 Ki > 100000 nM T94033 CS2D1R 44364505 Ki > 100000 nM T94033 CQE3K8 44364506 Ki = 13000 nM T94033 CT10GM 44364862 Ki > 5000 nM T94033 CDIR32 44364938 Ki > 5000 nM T94033 CL1O0R 44364939 Ki > 5000 nM T94033 CYD1M4 44364940 Ki > 5000 nM T94033 CXD05A 44364941 Ki > 5000 nM T94033 COJ03I 44364946 Ki > 5000 nM T94033 C5M2CT 44364948 Ki > 5000 nM T94033 CM87YB 44364952 Ki > 5000 nM T94033 CD93ET 44364982 Ki > 5000 nM T94033 CG4RV3 44364999 Ki > 5000 nM T94033 CTVZ78 44365103 Ki > 5000 nM T94033 CNO4X7 44365111 Ki > 5000 nM T94033 CIDS76 44365112 Ki > 5000 nM T94033 C4OE2C 44365192 Ki > 5000 nM T94033 CEH1M4 44365200 Ki > 5000 nM T94033 CFZ2T9 44365277 Ki > 5000 nM T94033 C3GA5J 44365287 Ki > 5000 nM T94033 CN4D2F 44365289 Ki > 5000 nM T94033 C5YT9W 44366105 Ki = 1400 nM T94033 CT1F2W 44366339 Ki = 1500 nM T94033 CKE86T 44366490 IC50 = 14000 nM T94033 C25DVX 44366493 IC50 = 2000 nM T94033 C6GU2Z 44366674 IC50 = 46000 nM T94033 C6TIQ1 44366772 IC50 = 8.6 nM T94033 C4UR5N 44366784 IC50 = 3 nM T94033 CWM1Q0 44366789 IC50 = 730 nM T94033 CWB84I 44366807 IC50 = 820 nM T94033 C2A7TO 44366810 IC50 > 1000000 nM T94033 C2ZUD0 44366829 IC50 > 1000000 nM T94033 CTY52Z 44366924 IC50 = 2 nM T94033 C3DUE7 44366925 IC50 = 2300 nM T94033 C01GQT 44368278 IC50 > 10000 nM T94033 CJ4O0M 44368282 IC50 > 10000 nM T94033 C67DWF 44368293 IC50 > 10000 nM T94033 C78XDG 44368377 IC50 > 10000 nM T94033 C1LST9 44368378 IC50 > 10000 nM T94033 CC2F9Z 44368575 IC50 > 10000 nM T94033 C6OF4C 44368576 IC50 > 10000 nM T94033 C37ZDX 44368590 IC50 > 10000 nM T94033 CCN24M 44368609 IC50 > 10000 nM T94033 CBT5V7 44368623 IC50 > 10000 nM T94033 C3PHI0 44369086 Ki = 2000 nM T94033 CWK6U8 44369271 Ki = 300 nM T94033 C1HBT5 44369288 Ki = 120 nM T94033 C6XB0Y 44371477 Ki > 2100 nM T94033 C3T0PF 44372395 Ki > 6300 nM T94033 CAJ92B 44372499 Ki = 6000 nM T94033 CI32UH 44372518 Ki = 3600 nM T94033 C7I3HS 44372533 Ki = 2640 nM T94033 CJE89V 44372620 Ki > 6300 nM T94033 C39FZP 44372663 Ki = 15000 nM T94033 C9I0BE 44372667 Ki = 4000 nM T94033 CQLA75 44372683 Ki = 15000 nM T94033 CKFN05 44372724 Ki > 1000000 nM T94033 CTD36H 44372738 Ki = 170000 nM T94033 CI6MQ5 44372778 Ki = 16000 nM T94033 CUVD59 44372831 Ki > 21000 nM T94033 CBLZ18 44372833 Ki = 3200 nM T94033 CFH41R 44372839 Ki = 10000 nM T94033 C9COY7 44372840 Ki > 1000000 nM T94033 C34AWY 44372863 Ki = 230000 nM T94033 CZE15A 44372864 Ki = 11000 nM T94033 C7X5BE 44372865 Ki = 12 nM T94033 C2E6TP 44372889 Ki = 33000 nM T94033 CNOV-41 44372899 Ki = 600 nM T94033 C36XWM 44372903 Ki = 50 nM T94033 C3MX0H 44374677 Ki = 5700 nM T94033 C4HSA0 44374690 Ki = 4500 nM T94033 CJC73F 44374707 IC50 = 55000 nM T94033 CWD13R 44374708 IC50 = 1100 nM T94033 C2Y0SC 44375908 IC50 > 500000 nM T94033 C3C2XE 44375967 IC50 = 669 nM T94033 C69QAS 44375986 IC50 = 870 nM T94033 C34XTM 44375987 IC50 = 10000 nM T94033 CZVP71 44376028 IC50 = 267 nM T94033 CZA1N6 44376029 IC50 = 809 nM T94033 C58WMI 44376046 IC50 = 375 nM T94033 C74KVW 44376051 IC50 = 11000 nM T94033 C6SC3T 44376056 IC50 = 14000 nM T94033 C2NHP9 44376074 IC50 = 751 nM T94033 CE9N6S 44376077 IC50 = 2000 nM T94033 C6QTS8 44376079 IC50 = 417 nM T94033 CEKQ15 44376084 IC50 = 185 nM T94033 C9T2QI 44376089 IC50 = 38 nM T94033 CD0W7C 44376100 IC50 = 1000 nM T94033 CG78SI 44376101 IC50 = 7000 nM T94033 CG9KH1 44376121 IC50 = 5000 nM T94033 C23ZRU 44376219 IC50 = 17000 nM T94033 C5PH2E 44376249 IC50 = 4000 nM T94033 C0Y8QD 44376252 IC50 = 2000 nM T94033 CD03ZI 44376253 IC50 = 4000 nM T94033 CX98EC 44376254 IC50 = 4000 nM T94033 C1F2JZ 44376255 IC50 = 5000 nM T94033 C7BS3N 44376258 Ki = 0.00065 nM T94033 C63JEF 44376259 IC50 = 2000 nM T94033 C0Z9CS 44376264 IC50 = 2000 nM T94033 CSRZ57 44376273 IC50 = 7000 nM T94033 CCY74M 44376286 IC50 = 5000 nM T94033 CP9IY1 44376287 IC50 = 3000 nM T94033 C0S9XG 44376288 IC50 = 6000 nM T94033 COX13N 44376289 IC50 = 573 nM T94033 CNC7F4 44376290 IC50 = 3000 nM T94033 C6X7UG 44376311 IC50 = 792 nM T94033 C4TGW5 44376318 IC50 = 3000 nM T94033 C28ZIJ 44376322 IC50 = 8000 nM T94033 C51GPZ 44376323 IC50 = 60000 nM T94033 C5Y6JB 44376326 IC50 = 1000 nM T94033 CA59MK 44376327 IC50 = 134 nM T94033 C5R2PM 44376328 IC50 = 751 nM T94033 CDM65F 44376342 IC50 = 4000 nM T94033 C6R5AG 44376343 IC50 = 118 nM T94033 C8M2PZ 44376385 IC50 = 12000 nM T94033 CB87VR 44376416 IC50 = 719 nM T94033 C5VDG0 44376417 IC50 = 569 nM T94033 C1S5KV 44376423 IC50 = 138 nM T94033 CG64YQ 44376426 IC50 = 390 nM T94033 COAE61 44376427 IC50 = 2000 nM T94033 CXEG05 44376429 IC50 = 642 nM T94033 CP7CO4 44376432 IC50 = 2000 nM T94033 CT8KB1 44376468 IC50 = 220000 nM T94033 CI03DP 44376475 IC50 = 8 nM T94033 CUVH30 44376476 IC50 = 5000 nM T94033 CSW71I 44376504 Ki = 3100 nM T94033 C9SW1H 44376514 IC50 = 12000 nM T94033 CM75ZP 44376515 IC50 = 40000 nM T94033 C51GQP 44376523 Ki = 8500 nM T94033 CA7GW4 44376525 Ki = 26000 nM T94033 CHW87S 44376544 IC50 = 3000 nM T94033 C3DLJ9 44376572 IC50 = 4000 nM T94033 C1PK0O 44376651 Ki = 1740 nM T94033 CMT40Z 44376656 Ki = 61 nM T94033 CH3V9X 44376684 Ki = 130 nM T94033 CJBO94 44376700 IC50 = 200000 nM T94033 C3K7NA 44376701 IC50 = 12000 nM T94033 CKSV26 44376702 IC50 = 3000 nM T94033 CXZP98 44376712 Ki = 7940 nM T94033 CUFO93 44376713 Ki = 7940 nM T94033 C1Z3BF 44376731 IC50 = 150000 nM T94033 CEKG07 44376754 Ki = 1350 nM T94033 CQX98K 44376755 Ki = 2300 nM T94033 C2JKH1 44376756 Ki = 1900 nM T94033 C9YJ8G 44376870 Ki = 85 nM T94033 C2EG6R 44376898 Ki = 28 nM T94033 C0SVG5 44376924 Ki = 97200 nM T94033 C8ZM6P 44376938 Ki = 40 nM T94033 C8P5YZ 44376949 IC50 = 2000 nM T94033 C7JL9O 44376950 Ki = 15600 nM T94033 CO2I5Z 44376952 Ki = 3060 nM T94033 CR6X9B 44376988 Ki = 200 nM T94033 C4XJD0 44377015 IC50 = 2000 nM T94033 CQB2G9 44377016 IC50 = 325000 nM T94033 CZ6MJ4 44377137 Ki = 62 nM T94033 CO0UK2 44377158 Ki = 31700 nM T94033 C67UJR 44377275 Ki = 220 nM T94033 CZ6W0S 44377280 Ki = 163.5 nM T94033 CVS76R 44377281 Ki = 10.8 nM T94033 CI2GS0 44377287 IC50 > 2500 nM T94033 C2MNC3 44377299 Ki = 61 nM T94033 C4HU2G 44377300 Ki > 397 nM T94033 CKX32Z 44377301 Ki = 14.4 nM T94033 CWN74Q 44377302 Ki = 282.5 nM T94033 C7W2GD 44377304 IC50 = 1100 nM T94033 C6RA4Q 44377310 Ki = 85.7 nM T94033 CG0S9N 44377311 Ki = 0.6 nM T94033 C3MQ4V 44377317 Ki = 166.7 nM T94033 CD1Q9R 44377318 Ki = 23.8 nM T94033 CP0V6X 44377320 IC50 > 2500 nM T94033 C4KSG5 44377322 IC50 > 2500 nM T94033 CH1NM4 44377327 IC50 > 2500 nM T94033 CTP28F 44377331 IC50 > 2500 nM T94033 CN42TW 44377336 Ki = 71.4 nM T94033 CPE23W 44377369 Ki = 6.2 nM T94033 C30VGP 44377425 IC50 > 2500 nM T94033 C39PST 44377471 Ki = 0.95 nM T94033 C5Q1LA 44377475 Ki = 19.4 nM T94033 CVHL28 44377478 Ki = 0.54 nM T94033 CT0G2D 44377544 IC50 > 2500 nM T94033 CK6I3F 44377546 IC50 > 2500 nM T94033 CNUL43 44377548 IC50 > 2500 nM T94033 CZBJ51 44377550 IC50 > 2500 nM T94033 CHU5T4 44377558 IC50 = 352 nM T94033 CY23PW 44377568 Ki = 53.2 nM T94033 CU49MW 44377570 Ki = 39.5 nM T94033 C3I2GH 44377571 Ki = 92.9 nM T94033 CRAS42 44377572 Ki > 397 nM T94033 C1TVZ9 44377573 Ki = 9 nM T94033 CGM35H 44377590 Ki = 195.2 nM T94033 C3LE7S 44377608 Ki = 29.8 nM T94033 C7Y4QI 44377622 Ki = 19.4 nM T94033 CXLT41 44377644 Ki = 13.3 nM T94033 CX5SE9 44377646 Ki = 239.7 nM T94033 CY1BO4 44378264 Ki = 0.3 nM T94033 CAH46S 44378457 Ki = 3.1 nM T94033 CD0M5Y 44378458 Ki = 24 nM T94033 CO7N6Y 44378546 Ki = 12900 nM T94033 CR8S2Q 44378621 Ki = 1.5 nM T94033 C3N7QV 44378628 Ki = 4.1 nM T94033 C1WB3Q 44378759 Ki = 12800 nM T94033 CLXH02 44378887 Ki = 289000 nM T94033 CGL17Z 44379037 Ki = 18 nM T94033 COH45E 44379112 Ki = 3.7 nM T94033 CMW49N 44379117 Ki = 3.2 nM T94033 CDW7T0 44379762 Ki = 52 nM T94033 C16RCS 44379766 Ki = 16 nM T94033 C05LCN 44379767 Ki = 44 nM T94033 C0KJW7 44379768 Ki = 3700 nM T94033 C9R0BW 44379807 Ki = 36 nM T94033 CUMV41 44379815 Ki = 445 nM T94033 C6IRM4 44379833 Ki = 190 nM T94033 CVZ62K 44379834 Ki = 35 nM T94033 C58QXF 44379842 Ki = 39 nM T94033 CS87LJ 44379843 Ki = 28 nM T94033 CIV0M9 44379856 Ki = 399 nM T94033 CY74CH 44379858 Ki = 327 nM T94033 CWJ5E6 44379904 Ki = 11 nM T94033 CJ0P4F 44379905 Ki = 0.33 nM T94033 CN1H0Z 44379935 Ki = 490 nM T94033 CMLO53 44379937 Ki = 30 nM T94033 CN29VI 44379953 Ki = 32 nM T94033 C9OX3G 44379960 Ki = 14 nM T94033 CY4HT3 44380201 Ki = 12 nM T94033 CI39WG 44380233 Ki = 22 nM T94033 CJ7ID6 44380246 Ki = 32 nM T94033 C9FWM3 44380247 Ki = 115 nM T94033 CGJ29X 44380265 Ki = 39 nM T94033 CD36KV 44380417 Ki = 0.0025 nM T94033 CI4RX8 44380662 IC50 = 44 nM T94033 CVG5S6 44380663 IC50 < 1 nM T94033 CC4MP1 44380667 Ki = 1.7 nM T94033 CC8DX1 44380674 IC50 = 340 nM T94033 CU98BT 44380699 IC50 = 15 nM T94033 CZ6NT9 44380722 IC50 = 18 nM T94033 C91WQC 44380740 IC50 = 2050 nM T94033 CUMQ41 44380741 IC50 = 750 nM T94033 C2XH6Q 44381062 IC50 = 57 nM T94033 C3I2DC 44381063 IC50 = 450 nM T94033 C8I5OP 44381104 IC50 = 77 nM T94033 CN5A4R 44381155 Ki = 2100 nM T94033 C5XC2T 44381273 Ki = 110 nM T94033 CJ6M5B 44382389 IC50 = 256 nM T94033 CTF4N6 44382391 IC50 = 50.5 nM T94033 CAI65F 44382441 IC50 = 472 nM T94033 C6LH5V 44383081 IC50 = 6.2 nM T94033 C9SD3E 44383242 Ki > 4000 nM T94033 C5PW9E 44383425 IC50 = 203 nM T94033 C43KTU 44383519 Ki > 4000 nM T94033 CNBG48 44383542 IC50 = 194 nM T94033 C2IX5U 44383543 IC50 = 89.1 nM T94033 C84TXN 44383800 Ki = 19 nM T94033 CBN31W 44384237 Ki > 21000 nM T94033 C5DAB6 44384238 Ki = 140 nM T94033 CE5P9W 44384391 Ki = 7.4 nM T94033 C6IX3V 44384674 Ki = 570 nM T94033 CP74XU 44384744 Ki = 5000 nM T94033 CGI1H8 44384745 Ki = 5000 nM T94033 CHK87Y 44384746 Ki = 490 nM T94033 CR2VG0 44384747 Ki = 98 nM T94033 CUR5K2 44384798 Ki > 5000 nM T94033 CQ1D0K 44384799 Ki > 5000 nM T94033 CNB73E 44384879 Ki = 28 nM T94033 C6H0NF 44384928 Ki = 7 nM T94033 CVYI62 44385066 Ki = 2670 nM T94033 CJ01YE 44385090 Ki = 2350 nM T94033 CV4N1P 44385091 Ki = 1050 nM T94033 C1ZV8A 44385092 Ki = 360 nM T94033 COQ8S6 44385134 Ki = 2700 nM T94033 CVGJ91 44385135 Ki = 5000 nM T94033 CLWT03 44385136 Ki = 4600 nM T94033 CT42KF 44385150 Ki = 650 nM T94033 CALR98 44385151 Ki = 300 nM T94033 CNH87R 44385152 Ki = 5000 nM T94033 C43MAX 44385153 Ki = 4610 nM T94033 CDT45B 44385195 Ki = 70 nM T94033 C7U0HZ 44385205 Ki = 520 nM T94033 CTX13E 44385259 Ki = 3530 nM T94033 CI91SG 44385260 Ki = 210 nM T94033 C4RV6U 44385263 Ki = 50 nM T94033 CNMA50 44385268 Ki = 5000 nM T94033 C3DF2V 44385269 Ki = 5000 nM T94033 C9Z1OC 44385301 Ki = 160 nM T94033 CHPL94 44385310 Ki = 4530 nM T94033 C6VZ5Y 44385361 Ki = 3780 nM T94033 CCR46P 44385364 Ki > 5000 nM T94033 CPV5B7 44385418 Ki = 4000 nM T94033 C8CE6A 44385432 Ki = 2320 nM T94033 CG7LT1 44385488 IC50 > 11000 nM T94033 C94GZU 44385541 IC50 > 11000 nM T94033 C3T9XK 44385607 IC50 > 11000 nM T94033 CKY0P4 44385611 IC50 > 11000 nM T94033 CUS20V 44385673 IC50 > 11000 nM T94033 CZ8XL6 44385679 IC50 > 11000 nM T94033 CL5BA4 44385729 IC50 > 11000 nM T94033 C3DSN7 44385768 IC50 > 11000 nM T94033 C8USN9 44385769 IC50 > 11000 nM T94033 C2E8DS 44385771 IC50 > 11000 nM T94033 C2VFC6 44385772 IC50 > 11000 nM T94033 CN8V0W 44385779 IC50 > 11000 nM T94033 CIHV71 44385786 Ki = 2000 nM T94033 CPOS98 44385789 Ki = 2400 nM T94033 C2WYO3 44385799 Ki = 810 nM T94033 CJ5B9H 44385803 Ki = 6000 nM T94033 CBEA65 44385842 IC50 > 11000 nM T94033 CN5Q1G 44385864 Ki = 870 nM T94033 C4XY8T 44385865 Ki = 1990 nM T94033 CC9M7E 44385869 IC50 > 11000 nM T94033 C8WK4A 44385891 IC50 > 11000 nM T94033 C42JCS 44385915 Ki = 950 nM T94033 C3D2CL 44385935 IC50 > 11000 nM T94033 CX1C3I 44385963 Ki = 2300 nM T94033 CFPH43 44385967 Ki = 170 nM T94033 CW08OY 44385998 IC50 > 11000 nM T94033 CV6KG4 44386059 IC50 > 11000 nM T94033 CWR4Q6 44386101 Ki = 3900 nM T94033 CJ48AC 44386102 Ki = 590 nM T94033 CGU69V 44386179 IC50 > 11000 nM T94033 CS65LH 44386185 IC50 > 11000 nM T94033 CU0P5T 44386242 IC50 > 11000 nM T94033 CU9J0D 44386250 IC50 > 11000 nM T94033 C9G7QW 44386322 IC50 > 11000 nM T94033 C31CUG 44386326 IC50 > 11000 nM T94033 CX58AM 44386358 Ki = 230 nM T94033 C2WCE4 44386371 IC50 > 11000 nM T94033 C52POK 44386417 IC50 > 11000 nM T94033 CRX1I9 44386418 IC50 > 11000 nM T94033 CIBD76 44386484 IC50 > 11000 nM T94033 C8ME4O 44386493 IC50 > 11000 nM T94033 CD4AH3 44386540 IC50 > 11000 nM T94033 CHAO48 44386542 IC50 > 11000 nM T94033 CLNO15 44386637 IC50 > 11000 nM T94033 C81IMH 44386642 IC50 > 11000 nM T94033 C4JB0M 44386841 IC50 > 11000 nM T94033 C5MR1F 44386934 IC50 > 11000 nM T94033 CA45DZ 44387044 IC50 > 11000 nM T94033 C39LUW 44387104 IC50 > 11000 nM T94033 C2QD1K 44387206 IC50 > 11000 nM T94033 C6SV1C 44387258 IC50 = 350 nM T94033 CR57NJ 44387819 IC50 = 17000 nM T94033 CAN0S2 44387823 Ki = 2.1 nM T94033 C6FTY4 44387829 Ki = 3.1 nM T94033 C3GO6F 44387834 Ki = 2400 nM T94033 CFD2J0 44387835 IC50 = 4.5 nM T94033 C6RB2U 44387843 IC50 = 5.3 nM T94033 CD0UY2 44387845 Ki = 2 nM T94033 CN2GR5 44390800 Ki = 540 nM T94033 CW3G5V 44390801 Ki = 6400 nM T94033 C7KZY2 44393000 Ki = 0.27 nM T94033 CX1FU9 44393017 Ki = 80 nM T94033 C1BC3J 44393086 Ki = 5.6 nM T94033 CZJ10X 44393132 Ki = 2.7 nM T94033 C60HBD 44393152 Ki = 4.7 nM T94033 CY6TW8 44393175 Ki = 0.5 nM T94033 CV3C5X 44393264 Ki = 0.9 nM T94033 CLM10G 44393633 IC50 > 10000 nM T94033 COS35W 44393635 IC50 > 10000 nM T94033 C54IJH 44393646 IC50 > 10000 nM T94033 C4J5YZ 44393648 IC50 > 10000 nM T94033 C7F1EZ 44393650 IC50 > 10000 nM T94033 CM15TG 44393671 IC50 > 10000 nM T94033 CW2B4G 44393673 IC50 > 10000 nM T94033 CAYT14 44393675 IC50 > 10000 nM T94033 CI7OZ9 44393679 IC50 > 10000 nM T94033 CO3B6P 44393688 IC50 > 10000 nM T94033 C5BWQ3 44393690 IC50 > 10000 nM T94033 CW7T2D 44393692 IC50 > 10000 nM T94033 CD0O9Q 44393694 IC50 > 10000 nM T94033 CU47SD 44393720 IC50 > 10000 nM T94033 C2Q6CA 44393722 IC50 > 10000 nM T94033 C95LDV 44393724 IC50 > 10000 nM T94033 C78QJO 44394249 Ki > 50000 nM T94033 CQRB69 44394250 Ki > 50000 nM T94033 CJ45KG 44395699 IC50 > 10000 nM T94033 CN04TX 44395725 IC50 > 10000 nM T94033 CN7Y2C 44395728 IC50 > 10000 nM T94033 C81TGP 44395751 IC50 > 10000 nM T94033 CS7UY1 44395771 IC50 > 10000 nM T94033 COD05Q 44395835 IC50 > 10000 nM T94033 CA0ZU3 44395871 IC50 > 10000 nM T94033 C1G7ZQ 44395885 IC50 > 10000 nM T94033 CIB17E 44395901 IC50 > 10000 nM T94033 C4SUD5 44396124 IC50 > 10000 nM T94033 CCL3J1 44396183 IC50 > 10000 nM T94033 CEC5X2 44396195 IC50 > 10000 nM T94033 CZ6S5M 44399310 Ki = 3.1 nM T94033 C62ZMT 44399434 Ki = 0.55 nM T94033 CL92RW 44399452 Ki = 0.77 nM T94033 CJO5L3 44399529 Ki = 550 nM T94033 CE5S0J 44400525 IC50 > 10000 nM T94033 CB0N5T 44400527 Ki > 100000 nM T94033 CH9TP3 44402039 Ki = 486 nM T94033 C49CME 44402191 Ki > 5000 nM T94033 CUB28Z 44402339 Ki = 260 nM T94033 C1TF0I 44402340 Ki = 20 nM T94033 CN76WZ 44402361 Ki = 150 nM T94033 CL80DH 44402364 Ki = 2507 nM T94033 CKTZ36 44402382 Ki = 0.48 nM T94033 CQ4J2A 44402383 Ki > 5000 nM T94033 C8WR3I 44402428 Ki > 5000 nM T94033 CJQ8X6 44402429 Ki = 4764 nM T94033 C6CZ8H 44402442 Ki = 500 nM T94033 CWK5D3 44402498 Ki = 3.2 nM T94033 CPLF17 44402521 Ki > 5000 nM T94033 C08ZRI 44402527 Ki = 0.45 nM T94033 C5JK1T 44402528 Ki > 5000 nM T94033 C9CWT3 44402591 Ki = 1682 nM T94033 CV0S6N 44402617 Ki = 1196 nM T94033 CTS5W9 44404049 IC50 > 400000 nM T94033 CRH8Z4 44404152 Ki = 0.08 nM T94033 C4F8BL 44404188 Ki = 9.4 nM T94033 CK13IB 44404219 Ki = 2.1 nM T94033 CU2R3Q 44406384 Ki = 53 nM T94033 CEM0T2 44406385 Ki = 6.4 nM T94033 CG06DH 44406389 Ki = 22 nM T94033 CYI68A 44406396 Ki = 380 nM T94033 CPD9E8 44406402 Ki = 350 nM T94033 CS2MJ9 44406408 Ki = 170 nM T94033 C1LUS7 44406409 Ki = 34 nM T94033 CL0QJ7 44406420 Ki = 198 nM T94033 CLUZ93 44406421 Ki = 30 nM T94033 CT1BO0 44406426 Ki = 65 nM T94033 CUDA42 44406438 Ki = 1800 nM T94033 C97JST 44406439 Ki = 10 nM T94033 C63USQ 44406471 Ki = 17 nM T94033 C43HWU 44406479 Ki = 450 nM T94033 CI3VX0 44406522 Ki = 6 nM T94033 CT13RQ 44406523 Ki = 2 nM T94033 CMP6S3 44406524 Ki = 200 nM T94033 CM0YG4 44406525 Ki = 193 nM T94033 CE07NJ 44406529 Ki = 143 nM T94033 CD3EI5 44406534 Ki = 1100 nM T94033 C40ESI 44407593 IC50 = 1100 nM T94033 CG3F5V 44407595 IC50 = 18000 nM T94033 CJT68D 44407597 IC50 = 2500 nM T94033 CH5L1B 44407599 IC50 = 1800 nM T94033 C6M0JA 44407601 IC50 = 1300 nM T94033 CLX0M1 44407607 IC50 = 1400 nM T94033 CMIF29 44407615 IC50 = 1600 nM T94033 CTC34S 44407621 IC50 = 4700 nM T94033 C70SUH 44407623 IC50 = 1900 nM T94033 C1G4BC 44407625 Ki = 320 nM T94033 CWUT14 44407627 IC50 = 120 nM T94033 CPM2L1 44407634 IC50 = 250 nM T94033 C5G7CN 44407639 IC50 = 130 nM T94033 CWE53V 44407641 IC50 = 190 nM T94033 CCQ4O8 44407688 IC50 = 3700 nM T94033 C0GV3X 44407749 IC50 = 25 nM T94033 C71VGN 44407751 IC50 = 82 nM T94033 C26PJY 44407814 IC50 = 670 nM T94033 C3GW8V 44407816 IC50 = 69000 nM T94033 C51QCV 44407822 IC50 = 970 nM T94033 C5VW4Y 44407825 IC50 = 2700 nM T94033 C4ZLJ0 44407830 IC50 = 16 nM T94033 CX79TB 44407832 IC50 = 39 nM T94033 CL1X5A 44407835 IC50 = 50 nM T94033 C0KAH8 44407838 IC50 = 97 nM T94033 C2E0JC 44407841 IC50 = 3100 nM T94033 C7QK8H 44407843 IC50 = 2100 nM T94033 C36OIS 44407846 IC50 = 4100 nM T94033 C3KTD2 44407848 IC50 = 1500 nM T94033 CS4C2A 44407852 IC50 = 2400 nM T94033 CY87PU 44407854 IC50 = 190 nM T94033 CEDS48 44407856 IC50 = 260 nM T94033 C6PVI3 44407859 IC50 = 590 nM T94033 CJ50KO 44407866 IC50 = 570 nM T94033 C4WPB9 44407868 IC50 = 1000 nM T94033 C6R2YO 44407889 IC50 = 15000 nM T94033 C1LUR9 44407946 IC50 = 3000 nM T94033 CVSE54 44407974 IC50 = 330 nM T94033 C9N1SL 44407977 IC50 = 340 nM T94033 C71TKS 44407986 IC50 = 3100 nM T94033 CK9YT6 44407994 IC50 = 20000 nM T94033 CDUS65 44407995 IC50 = 14000 nM T94033 CZ69GQ 44408053 IC50 = 810 nM T94033 CJ3P4D 44408067 IC50 = 170 nM T94033 C7NYX6 44409708 IC50 > 300000 nM T94033 CEGD74 44409709 IC50 = 284000 nM T94033 CM3U5W 44409710 IC50 > 300000 nM T94033 CZ97DT 44409713 IC50 = 48000 nM T94033 CQC74T 44409732 IC50 = 107000 nM T94033 C0G1MU 44409734 IC50 > 300000 nM T94033 CIKW90 44409735 IC50 = 151000 nM T94033 C79XCS 44409750 IC50 > 300000 nM T94033 C6V5KN 44409930 IC50 > 300000 nM T94033 CZ6O0S 44410963 IC50 = 44.2 nM T94033 CO56UV 44410975 IC50 = 56.3 nM T94033 CL1X5B 44410980 IC50 = 58.4 nM T94033 CFU4T2 44410981 IC50 = 16 nM T94033 C9JQ1N 44411024 IC50 = 31.9 nM T94033 CM97AD 44411055 IC50 = 76.8 nM T94033 CIWD48 44411064 IC50 = 53600 nM T94033 CNA17B 44411074 IC50 = 288 nM T94033 CY45TS 44411083 IC50 = 6.4 nM T94033 CP67EA 44411094 IC50 = 1.29 nM T94033 CYLC35 44411097 IC50 = 581 nM T94033 C1XFL2 44411136 IC50 = 44 nM T94033 CM8OZ0 44411137 IC50 = 1.76 nM T94033 C9U7FN 44411143 IC50 = 4.28 nM T94033 C0X1YL 44411144 IC50 = 9.88 nM T94033 CWO80X 44411151 IC50 = 50.9 nM T94033 CRS85H 44411152 IC50 = 33.9 nM T94033 C4N6VB 44411157 IC50 = 1080 nM T94033 C5WH8F 44411158 IC50 = 2780 nM T94033 C4WG8Q 44411164 IC50 = 566 nM T94033 C15XEK 44411242 IC50 = 3.4 nM T94033 CD6C1U 44411250 IC50 = 2.7 nM T94033 C8Z9VS 44411256 IC50 = 1430 nM T94033 CQ34JF 44411342 IC50 = 20.8 nM T94033 C4QFU7 44411350 IC50 = 71.2 nM T94033 CND8S5 44411365 IC50 = 103 nM T94033 CR2VW4 44411385 IC50 = 4090 nM T94033 C2C8OJ 44411386 IC50 = 49.1 nM T94033 C7VLB6 44411433 IC50 = 1020 nM T94033 C80CNW 44411436 IC50 = 2.15 nM T94033 CQ21SX 44411439 IC50 = 232 nM T94033 C1COF3 44411461 IC50 = 290 nM T94033 CB20AJ 44411467 IC50 = 14.8 nM T94033 CH4M0J 44411511 IC50 = 51.2 nM T94033 C58XZT 44411539 IC50 = 1370 nM T94033 CB1G3D 44412151 Ki = 1070 nM T94033 CC2Z1K 44412258 Ki > 100000 nM T94033 CLQ54S 44412280 Ki = 7900 nM T94033 C3BX5Y 44412781 Ki > 150000 nM T94033 CF5XO4 44413343 Ki = 13000 nM T94033 CTD42X 44413355 Ki = 170 nM T94033 C9KQM2 44413356 Ki = 1700 nM T94033 CQDX92 44413619 Ki = 1300 nM T94033 CO8A0Y 44414333 Ki = 48000 nM T94033 CO6Z9S 44415089 IC50 = 85000 nM T94033 CG6H0U 44415561 Ki = 100000 nM T94033 C3LCV6 44415581 Ki = 99000 nM T94033 CPN1S0 44416248 IC50 = 6000 nM T94033 CJ20PN 44416510 IC50 = 129000 nM T94033 CZK3N4 44416547 IC50 = 30800 nM T94033 CQA4B5 44416549 IC50 = 5500 nM T94033 CMVF02 44416571 IC50 = 12300 nM T94033 C3TJK6 44418750 IC50 = 6700 nM T94033 C7LK8E 44418751 IC50 = 4300 nM T94033 C9G1VL 44418752 IC50 = 2100 nM T94033 CHK10G 44418753 IC50 = 2100 nM T94033 C9OZ1M 44418754 IC50 = 935 nM T94033 CVJ85S 44421826 IC50 > 200000 nM T94033 CWVX31 44421837 IC50 > 200000 nM T94033 CD58ZY 44421845 IC50 > 200000 nM T94033 C48NZW 44426214 Ki = 2700 nM T94033 COUZ56 44426215 Ki = 88000 nM T94033 C3F2PN 44426216 Ki > 1000000 nM T94033 CZ91LH 44426217 Ki = 10000 nM T94033 CEV53U 44426218 Ki = 7600 nM T94033 C8O6HV 44426219 Ki = 170 nM T94033 CJH6E4 44426220 Ki = 40000 nM T94033 C3E2FT 44426221 Ki = 190000 nM T94033 CW3G0D 44426222 Ki = 140000 nM T94033 CN6VL5 44426224 Ki = 1005 nM T94033 CG9XF0 44426226 Ki = 930 nM T94033 CQ7CF9 44426227 Ki = 2700 nM T94033 CL4N6J 44426228 Ki = 530 nM T94033 CJ3B7D 44426229 Ki = 8300 nM T94033 C5Q8HB 44426230 Ki = 6500 nM T94033 C6RNO7 44426232 Ki = 18000 nM T94033 CCGR09 44426234 Ki = 40000 nM T94033 CD06OJ 44426235 Ki = 140000 nM T94033 CR4D0U 44426236 Ki = 125000 nM T94033 CIT7D5 44426237 Ki = 24 nM T94033 CW71LJ 44426238 Ki = 250 nM T94033 CY5Z6P 44426239 Ki = 860 nM T94033 CI0N7E 44426240 Ki = 180 nM T94033 C35VBM 44426241 Ki = 20000 nM T94033 C0LIG6 44426243 Ki = 0.56 nM T94033 C9V2JR 44426244 Ki = 7.7 nM T94033 C72TBW 44426245 Ki = 19 nM T94033 CZ2GS7 44426246 Ki = 17.7 nM T94033 CPKM97 44426247 Ki = 4.9 nM T94033 C1MVS4 44426248 Ki = 7.8 nM T94033 C5W1RJ 44426249 Ki = 9 nM T94033 C8H5OR 44426250 Ki = 17.3 nM T94033 C8BE9L 44426251 Ki = 3.8 nM T94033 CT6C5J 44426252 Ki = 3.5 nM T94033 CCN6T9 44426253 Ki = 3.6 nM T94033 C1UYG6 44426254 Ki = 3.2 nM T94033 CGV1I0 44426657 IC50 = 10600 nM T94033 CXI16J 44426658 IC50 = 12800 nM T94033 CZ9O0J 44426660 IC50 > 100000 nM T94033 CJN3M1 44426799 IC50 > 30000 nM T94033 CO9Q4B 44427316 IC50 > 30000 nM T94033 CD9O6E 44427319 IC50 > 30000 nM T94033 C53IBP 44428362 Ki = 3200 nM T94033 C1Q0EO 44429102 IC50 > 100000 nM T94033 CV7A9L 44429104 IC50 > 100000 nM T94033 CB27IK 44429106 IC50 > 100000 nM T94033 CH6Z7Y 44429108 IC50 > 100000 nM T94033 C8IHX6 44429109 IC50 > 100000 nM T94033 CO78JZ 44429110 IC50 > 100000 nM T94033 CVO5Q1 44432538 Ki = 3601 nM T94033 CQIX73 44434809 Ki > 12000 nM T94033 C5R8HJ 44434815 Ki > 12000 nM T94033 COG34X 44434818 Ki = 5440 nM T94033 C9T1DP 44434835 Ki = 3950 nM T94033 C4ADI5 44435823 Ki > 2500 nM T94033 C30CFX 44436704 IC50 = 780 nM T94033 CY74ON 44441049 IC50 = 220 nM T94033 C23AEP 44441050 IC50 = 120 nM T94033 C7FLO0 44441052 IC50 = 97 nM T94033 C1TIX2 44441055 IC50 = 1500 nM T94033 CMJD73 44441056 IC50 = 5600 nM T94033 CZ6EY2 44441057 IC50 = 310 nM T94033 CYR65V 44441060 IC50 = 1.6 nM T94033 CPVF51 44441061 IC50 = 3.3 nM T94033 C4V7OU 44441063 IC50 = 7 nM T94033 CUNK31 44441065 IC50 = 3.4 nM T94033 CKI79V 44441068 IC50 = 101 nM T94033 C53LQB 44441072 IC50 = 786 nM T94033 C21XJB 44441075 IC50 = 53 nM T94033 CQZ6A2 44441082 IC50 = 334 nM T94033 CQ3T8I 44441087 IC50 = 171 nM T94033 CR2X1Y 44441091 IC50 = 11 nM T94033 CHB06C 44441284 IC50 = 27000 nM T94033 C8WL7U 44441285 IC50 = 36000 nM T94033 CVIO95 44441287 IC50 > 100000 nM T94033 CB49OX 44441290 IC50 > 100 nM T94033 CK3FA1 44443550 Ki = 33.9 nM T94033 C9FO1U 44443551 Ki = 2.7 nM T94033 CQ45MH 44443553 Ki = 4.7 nM T94033 C4M6QI 44443554 Ki = 1281 nM T94033 C71OTV 44443555 Ki = 58 nM T94033 C0HK3X 44443556 Ki = 128 nM T94033 C4JZ2V 44443559 Ki = 8.6 nM T94033 CTP1D9 44443561 Ki = 169 nM T94033 C0H3BA 44443562 Ki = 1.8 nM T94033 C6LG9A 44443564 Ki = 57 nM T94033 CMW64B 44443565 Ki = 142 nM T94033 CJ97OZ 44443566 Ki = 0.9 nM T94033 CZTC23 44444412 Ki > 6300 nM T94033 CT0K6W 44444413 Ki > 20000 nM T94033 C2GQ4X 44444414 Ki = 19200 nM T94033 CFS7X6 44444905 Ki = 33 nM T94033 CHRX61 44445075 IC50 = 26300 nM T94033 C5WH9G 44446642 Ki = 350 nM T94033 CU3YD7 44446648 Ki = 310 nM T94033 CSR9L5 44446652 Ki > 21000 nM T94033 CH27CY 44446654 Ki > 21000 nM T94033 CNX71T 44446656 Ki > 6300 nM T94033 C8T7LJ 44446659 Ki > 15000 nM T94033 C4S8CN 44447557 IC50 = 91 nM T94033 CUX8V1 44447559 IC50 = 92 nM T94033 CMK2J4 44447561 IC50 = 307 nM T94033 C64AGC 44447563 IC50 = 578 nM T94033 C1T8IL 44447565 IC50 = 885 nM T94033 CPC74I 44447567 IC50 = 1050 nM T94033 C5MQ8H 44447569 IC50 = 1180 nM T94033 CY65RS 44447571 IC50 = 1243 nM T94033 CP31IQ 44447573 IC50 = 1846 nM T94033 CN38RY 44447575 IC50 = 1919 nM T94033 CYE09U 44447577 IC50 = 2470 nM T94033 C5ISZ3 44447579 IC50 = 2706 nM T94033 CK16ZS 44447581 IC50 = 3091 nM T94033 C3J7LH 44447583 IC50 > 44400 nM T94033 CU73PM 44447585 IC50 > 44400 nM T94033 CBO20E 44447587 IC50 > 44400 nM T94033 COP7I8 44447589 IC50 > 44400 nM T94033 CJZ3U5 44447590 IC50 > 44400 nM T94033 CA35UW 44447591 IC50 > 44400 nM T94033 C0A6SV 44447592 IC50 > 44400 nM T94033 CV5L7W 44447593 IC50 > 44400 nM T94033 CN3SD5 44448299 Ki = 1.2 nM T94033 C7TJ5Q 44448740 Ki = 0.38 nM T94033 C8PH9I 44453003 Ki = 0.2 nM T94033 CG6LH2 44453056 IC50 = 3700 nM T94033 CC6A4Y 44453083 IC50 = 68 nM T94033 C06BVN 44453135 IC50 = 200000 nM T94033 C94URG 44453211 IC50 = 40 nM T94033 C0L4EK 44453237 IC50 = 980 nM T94033 C41ZMA 44453261 Ki = 3 nM T94033 CYI3H5 44453262 Ki = 0.68 nM T94033 CNC85E 44453287 Ki = 0.3 nM T94033 C4MB5N 44453288 Ki = 0.31 nM T94033 CX7U8Y 44453318 Ki = 0.65 nM T94033 CA9U8Y 44453319 Ki = 0.9 nM T94033 C4D2EV 44453334 IC50 = 11000 nM T94033 CU3BS5 44453335 IC50 = 390 nM T94033 CBH4T0 44453339 IC50 = 1200 nM T94033 CVGH52 44453355 Ki = 2.4 nM T94033 C67LIT 44453358 Ki = 2.8 nM T94033 C2SH5L 44453374 IC50 = 7000 nM T94033 CSC10P 44453375 IC50 = 420 nM T94033 CVJ75F 44453398 Ki = 1.9 nM T94033 C0U3TE 44453410 IC50 = 14000 nM T94033 C3D4NI 44453431 Ki = 0.19 nM T94033 CE86KR 44453432 Ki = 0.83 nM T94033 CVM4X7 44453434 Ki = 1.1 nM T94033 C0V3FO 44453445 IC50 = 38 nM T94033 CLGY91 44453465 Ki = 1.8 nM T94033 CN65UR 44453506 IC50 = 19000 nM T94033 CSFD95 44453524 Ki = 2 nM T94033 C9FI7C 44453526 Ki = 0.36 nM T94033 C1NM4O 44453556 Ki = 0.48 nM T94033 C6WGH0 44453588 IC50 = 1000 nM T94033 CV7FC4 44453589 IC50 = 5000 nM T94033 C7RNB9 44453659 Ki = 18 nM T94033 C5QIN2 44453660 Ki = 10 nM T94033 C72DAM 44453661 Ki = 24 nM T94033 CW1GP4 44453663 IC50 = 51 nM T94033 CHY5U4 44453679 Ki = 16 nM T94033 CW6D8F 44453680 Ki = 1 nM T94033 C4L6GX 44453709 Ki = 5 nM T94033 CVI9A6 44453803 Ki = 18 nM T94033 C7BJ0U 44453806 Ki = 2600 nM T94033 CPK79S 44453883 IC50 < 1 nM T94033 CS7BK4 44453888 Ki = 400 nM T94033 C8ZYV5 44453904 IC50 = 2370 nM T94033 COH2W3 44454019 Ki = 500 nM T94033 CTF95R 44454022 Ki = 65 nM T94033 CBA96S 44457762 IC50 = 4000 nM T94033 C4N7KR 44457766 IC50 = 84000 nM T94033 C6TFX8 44457896 Ki = 60 nM T94033 C2VAB4 44457926 Ki = 8700 nM T94033 C0Q7OB 44457944 IC50 = 22 nM T94033 CPXA19 44457985 Ki = 4.9 nM T94033 C3H9RE 44458036 Ki = 68 nM T94033 COE83M 44458061 Ki = 8.8 nM T94033 C0GCJ3 44458084 Ki = 97 nM T94033 CB4P1V 44458141 Ki = 1.6 nM T94033 C3B0TA 44458142 Ki = 570 nM T94033 CWS61M 44458143 Ki = 59 nM T94033 C5Z9CS 44458144 Ki = 7400 nM T94033 CA2ZK4 44458145 Ki = 120 nM T94033 C4DE1S 44458177 IC50 = 12000 nM T94033 C1DBQ3 44458182 Ki = 50 nM T94033 CH4IG1 44459090 Ki = 2000 nM T94033 CV5TB1 44459377 Ki = 10000 nM T94033 CVBZ10 44459392 Ki = 1500 nM T94033 CGS82Z 44459487 Ki = 120000 nM T94033 C95MDP 44459488 Ki = 200 nM T94033 CJ16HT 44459496 Ki = 300000 nM T94033 CZC3P9 44459497 Ki = 30000 nM T94033 CS1TF7 44460215 IC50 = 14.9 nM T94033 CVU5G4 44460232 IC50 = 137.5 nM T94033 CH61KG 44460246 IC50 = 125 nM T94033 C8SC7A 44460306 IC50 = 2.07 nM T94033 CXG8H0 44460987 Ki = 90 nM T94033 CO4PE2 44461072 Ki = 15 nM T94033 C8XDY2 44461086 IC50 = 12589.25 nM T94033 C5KH3T 44461169 IC50 = 12589.25 nM T94033 CBX36G 44461172 IC50 = 12589.25 nM T94033 C9BY7A 44461270 IC50 = 12589.25 nM T94033 CTCQ50 44461663 Ki = 0.7 nM T94033 CA2PX7 44461750 Ki = 0.2 nM T94033 CJ7SV4 44461896 Ki = 825 nM T94033 CWND94 44461897 IC50 = 370 nM T94033 CZ1YR4 44461912 Ki = 30 nM T94033 CK3F7D 44461986 Ki = 0.2 nM T94033 C13ZYL 44461991 Ki = 105 nM T94033 CX2LS5 44461992 IC50 = 750 nM T94033 C38UKJ 44461994 Ki = 75 nM T94033 C8Y7IF 44461995 Ki = 165 nM T94033 CF0N9S 44461996 Ki = 98 nM T94033 CH87SR 44462009 Ki = 1.8 nM T94033 CPY92L 44462032 IC50 = 280 nM T94033 C74KGD 44462047 Ki = 495 nM T94033 C8BH4N 44462081 IC50 = 137.5 nM T94033 CL1TX8 44462086 IC50 = 210 nM T94033 CXMW10 44462102 IC50 = 110 nM T94033 C0K9TY 44462103 IC50 = 210 nM T94033 CH3WY6 44462136 Ki = 40 nM T94033 CA8K6V 44462137 Ki = 43 nM T94033 C1B5XA 44462146 IC50 = 240 nM T94033 C74CRB 44462147 Ki = 80 nM T94033 C2UR1M 44462161 Ki = 20 nM T94033 CQ31TR 44462179 IC50 = 350 nM T94033 CU8Q5J 44462244 Ki = 55 nM T94033 C2SOP1 44462250 IC50 = 1000 nM T94033 C9Y8EN 44462296 IC50 = 1230 nM T94033 C1LG0F 44462297 IC50 = 990 nM T94033 CWB04E 44462312 IC50 = 64.4 nM T94033 CS84NF 44462330 Ki = 8 nM T94033 CT6S5P 44462346 IC50 = 3400 nM T94033 C5GR0E 44462347 Ki = 32 nM T94033 CDN1P2 44462348 IC50 = 250 nM T94033 CVZW52 44537923 IC50 = 4 nM T94033 C97LMR 44555350 IC50 = 3 nM T94033 C0UC8T 44567656 Ki = 500 nM T94033 CBJ1W7 44567658 Ki = 360 nM T94033 CP2FZ0 44567660 Ki = 57 nM T94033 CQYZ04 44567683 Ki = 310 nM T94033 CEW6G1 44569299 Ki = 520 nM T94033 C9JNT3 44569300 Ki = 310 nM T94033 C9XE7Q 44569301 Ki > 1000000 nM T94033 CZI8D7 44569333 Ki = 325000 nM T94033 CR4CP6 44569359 Ki = 9800 nM T94033 C9JF7W 44569667 Ki = 460 nM T94033 C61IJB 44569732 Ki = 2200 nM T94033 CR36MB 44569733 Ki = 5500 nM T94033 CE25UL 44569767 Ki = 1900 nM T94033 C0CZ4I 44569768 Ki = 1200 nM T94033 CIR4M0 44569769 Ki = 56 nM T94033 C02SHD 44569811 Ki = 11 nM T94033 CG3LE9 44569812 Ki = 51 nM T94033 CCU7V0 44569813 Ki = 10 nM T94033 C8BR6E 44569843 Ki = 450 nM T94033 C7Q9BH 44569844 Ki = 240 nM T94033 CZ35OW 44569845 Ki = 1100 nM T94033 CHV9C1 44569846 Ki = 33 nM T94033 C5JQ4W 44569889 Ki = 160 nM T94033 CE1O4I 44569890 Ki = 150 nM T94033 C4JU7I 44569891 Ki = 190 nM T94033 CGS83Z 44569892 Ki = 110 nM T94033 C4BN3H 44573109 Ki = 850 nM T94033 COR57Y 44573272 Ki = 110 nM T94033 C6DX3Y 44573273 Ki = 350 nM T94033 CM2R1P 44573274 Ki = 29000 nM T94033 CSP1I0 44573310 Ki = 14500 nM T94033 C6EG9V 44573311 Ki = 2300 nM T94033 CYV3X2 44573378 Ki = 395 nM T94033 CWUA41 44573379 Ki = 24200 nM T94033 CYA64G 44573380 Ki = 10600 nM T94033 CLG42S 44573428 Ki = 159000 nM T94033 C85KLF 44575432 IC50 > 100 ug.mL-1 T94033 CI20LY 44575435 IC50 = 27 ug.mL-1 T94033 CK62HU 44575438 IC50 = 35 ug.mL-1 T94033 CO9TB6 44575439 IC50 = 9 ug.mL-1 T94033 CZ2EC1 44575441 IC50 = 25 ug.mL-1 T94033 C0PMW3 44584374 Ki > 5100 nM T94033 CR6X5Q 44587208 Ki = 500 nM T94033 C87KXE 44587209 Ki = 150 nM T94033 C94YMX 44587229 Ki = 13342 nM T94033 C09ROK 44587230 Ki = 3362 nM T94033 CGOR19 44587231 Ki = 220 nM T94033 C8WH9R 44587232 Ki = 55 nM T94033 C3WOP7 44587261 Ki = 3400 nM T94033 CX1DP6 44587262 Ki = 760 nM T94033 C7K6JN 44587263 Ki = 5490 nM T94033 CKL1J2 44587264 Ki = 5731 nM T94033 CTF79D 44587290 Ki = 680 nM T94033 CBXY02 44587291 Ki = 45500 nM T94033 CDBV80 44587292 Ki = 25300 nM T94033 CWZ34J 44587314 Ki = 3850 nM T94033 CI51KQ 44587315 IC50 = 88 nM T94033 C1LR3H 44587316 IC50 = 10000 nM T94033 CN2A1O 44587317 IC50 = 83000 nM T94033 CI5C1F 44592560 IC50 = 12.98 nM T94033 CHK9G2 44592562 IC50 = 22.73 nM T94033 CNIX06 44592593 IC50 = 56.22 nM T94033 CZJ7C6 44592617 IC50 = 39.57 nM T94033 C1A8YB 44592658 IC50 = 50 nM T94033 CN7G0O 44592693 IC50 = 50 nM T94033 CC65UK 44592729 IC50 = 14.67 nM T94033 C9OG6N 44592765 IC50 = 86.86 nM T94033 CKC2Q8 44592831 IC50 = 63.1 nM T94033 CY2IM4 44592833 IC50 = 156.8 nM T94033 CW72YN 44592864 IC50 > 50 nM T94033 CD4G2B 44592865 IC50 > 50 nM T94033 CDLY78 44592888 IC50 = 8.51 nM T94033 C4RDW0 44592955 IC50 = 50 nM T94033 C1PLT5 44592978 IC50 = 12.3 nM T94033 CVS21G 44592979 IC50 = 50.24 nM T94033 C4M0KI 44593006 IC50 = 17.9 nM T94033 C9PCO6 44593008 IC50 = 4.88 nM T94033 C18VRK 44603851 IC50 = 570 nM T94033 C2PVE0 45103523 Ki = 2.3 nM T94033 CGN14R 45103723 Ki = 1.7 nM T94033 CCT47Y 45139983 Ki = 3810 nM T94033 CT6AS0 45139985 Ki = 940 nM T94033 CIJ1M2 45139988 Ki = 1640 nM T94033 CP1UO0 45140189 Ki = 3610 nM T94033 CBXF78 45140570 Ki = 1420 nM T94033 CCD71S 45140573 Ki = 70 nM T94033 C3FSP8 45140765 Ki = 150 nM T94033 C6G3WT 45140768 Ki = 11 nM T94033 CDK64S 45140770 Ki = 23 nM T94033 CE9NQ1 45141147 Ki = 1460000 nM T94033 C9P0GA 45141148 Ki = 330000 nM T94033 CX51QE 45141149 Ki = 322000 nM T94033 C09XHS 45141150 Ki = 155000 nM T94033 C04WFG 45141151 Ki = 484000 nM T94033 CVCY39 45141359 Ki = 72400 nM T94033 CV6S0C 45141360 Ki = 34500 nM T94033 C1SJ8Q 45141361 Ki = 92900 nM T94033 CFP10G 45141362 Ki = 29700 nM T94033 C2GM1T 45141363 Ki = 28000 nM T94033 CHIG82 45141792 Ki = 8080 nM T94033 C7C0XP 45141794 Ki = 33000 nM T94033 CY73JH 45142000 Ki = 2540 nM T94033 C6KIQ3 45142002 Ki = 920 nM T94033 CMUK63 45142003 Ki = 1300 nM T94033 CU9EB0 45142005 Ki = 410 nM T94033 C6R7DO 45142007 Ki = 430 nM T94033 CD3I5J 45142009 Ki = 40 nM T94033 CUQF60 45261201 IC50 = 270 nM T94033 CEXO72 45261244 IC50 = 110 nM T94033 CZ4JW1 45261445 Ki = 2000 nM T94033 C21DFE 45261835 Ki = 24 nM T94033 C3P8EA 45263195 IC50 > 10000 nM T94033 CK7E3M 45264760 Ki = 3600 nM T94033 CLD8H2 45265181 Ki = 47 nM T94033 C0SG1F 45266989 IC50 = 33000 nM T94033 C5E6AS 45267012 IC50 = 10000 nM T94033 CGF36S 45267239 IC50 = 0.57 ug.mL-1 T94033 CONF35 45267242 IC50 = 0.65 ug.mL-1 T94033 CWH6C4 45267245 IC50 = 0.43 ug.mL-1 T94033 C4SZR2 45267833 IC50 = 130000 nM T94033 CGU67A 45267836 IC50 = 33000 nM T94033 CW3SX0 45267838 IC50 = 33000 nM T94033 CG1OB3 45268701 IC50 > 33000 nM T94033 C2E6TJ 45268705 IC50 = 88000 nM T94033 CY75OX 45268711 IC50 = 790 nM T94033 CI64KY 45268962 IC50 = 1.5 ug.mL-1 T94033 CQ1BJ6 45268971 IC50 = 0.43 ug.mL-1 T94033 CT6AE1 45269564 IC50 = 100000 nM T94033 CSY60N 45269572 IC50 = 10000 nM T94033 CM2A6I 45269821 IC50 = 0.092 ug.mL-1 T94033 C2GM1C 45269827 IC50 = 3.5 ug.mL-1 T94033 CN70AY 45269834 IC50 = 0.28 ug.mL-1 T94033 COA86N 45270402 IC50 = 1890 nM T94033 CFQ14D 45270405 IC50 = 10000 nM T94033 CH1P5M 45270407 IC50 = 6230 nM T94033 CR36LB 45270649 IC50 = 3 ug.mL-1 T94033 CFNC61 45270659 IC50 = 0.2 ug.mL-1 T94033 C23ASP 45270664 IC50 = 0.03 ug.mL-1 T94033 CN5RH1 45270665 IC50 = 10 ug.mL-1 T94033 CU26GQ 45271227 IC50 = 7050 nM T94033 C68PDT 45271471 IC50 = 0.62 ug.mL-1 T94033 CLD09N 45271484 IC50 = 0.41 ug.mL-1 T94033 CQX07L 45272124 IC50 = 133000 nM T94033 CW6CB5 45272126 IC50 = 33000 nM T94033 C4P3OE 45272377 IC50 = 0.5 ug.mL-1 T94033 CTR67K 45272950 IC50 = 87000 nM T94033 CM9Y1C 45272953 IC50 = 300000 nM T94033 CJC3U4 45272961 IC50 = 88000 nM T94033 C58IBS 45273261 IC50 = 0.05 ug.mL-1 T94033 CNS6X8 45379634 IC50 = 52900 nM T94033 CJ73BT 45486346 Ki = 102000 nM T94033 C9ETC4 45486354 Ki = 50000 nM T94033 C73QKO 45486757 IC50 = 241 nM T94033 C2KR5T 45486768 IC50 = 11 nM T94033 C18IRX 45486770 IC50 = 44 nM T94033 C5E7FM 45486774 IC50 = 10 nM T94033 CE4M2H 45486784 IC50 = 106 nM T94033 C3S6QI 45486788 IC50 = 6 nM T94033 CH81PN 45486811 IC50 = 3960 nM T94033 C51ARS 45486812 IC50 = 3.3 nM T94033 CPYG61 45486813 IC50 = 3.4 nM T94033 CCG5U1 46196561 Ki = 1900 nM T94033 CD4T1L 46221636 IC50 = 92000 nM T94033 CZS2I0 46228551 Ki = 540 nM T94033 CKW04B 46228616 Ki = 1280 nM T94033 CSB71X 46228663 Ki = 20 nM T94033 C4YAJ7 46228924 IC50 > 100000 nM T94033 CW47XK 46232635 Ki > 21000 nM T94033 C62RBC 46835135 Ki > 25000 nM T94033 CY47OV 46878192 Ki = 43 nM T94033 C46KJA 46878193 Ki = 150 nM T94033 CQ2G6A 46878194 Ki = 2.1 nM T94033 C39CXL 46878195 Ki = 2000 nM T94033 C2VMH6 46878196 Ki = 8.8 nM T94033 CC6GE9 46878197 Ki = 3.2 nM T94033 CE79OB 46878198 Ki = 199 nM T94033 CS07EW 46878199 Ki = 507 nM T94033 C3HZP7 46878200 Ki = 67 nM T94033 CF5ZQ8 46878201 Ki = 15 nM T94033 C7ICJ0 46878202 Ki = 650 nM T94033 CQJR51 46878203 Ki = 0.04 nM T94033 C9BXU7 46878204 Ki = 350 nM T94033 CXQL63 46878205 Ki = 600 nM T94033 CR93NC 46878206 Ki = 230 nM T94033 C0H3UO 46878241 Ki > 5000 nM T94033 CO05NA 46881046 IC50 = 45200 nM T94033 C65OUI 46881272 Ki = 37 nM T94033 C4RSI0 46899736 Ki = 0.102 nM T94033 CX0Y2G 46899738 Ki = 0.052 nM T94033 CM90YX 46905275 Ki = 0.003 nM T94033 C6UNR5 46905276 Ki = 0.005 nM T94033 C8UXT3 46905277 Ki = 0.003 nM T94033 C2IXJ0 46905278 Ki = 0.015 nM T94033 CF24YP 46905279 Ki = 0.045 nM T94033 CW06NQ 46905280 Ki = 0.044 nM T94033 C01RYE 46905281 Ki = 0.1 nM T94033 CO9DV2 46905282 Ki = 0.036 nM T94033 C15YNV 46905283 Ki = 0.16 nM T94033 CH3J0U 46905284 Ki = 0.036 nM T94033 C7WC8Q 46905314 IC50 = 3.6 nM T94033 CNA06P 46905365 Ki = 2200 nM T94033 CNVR31 46905372 IC50 = 380 nM T94033 CX2L8G 46905375 Ki = 2400 nM T94033 CTR32W 46905376 Ki = 500 nM T94033 CS8GZ7 46905377 Ki = 6800 nM T94033 C9W1ZK 46905378 Ki = 5300 nM T94033 CR6P1E 46905379 Ki = 6300 nM T94033 CEDL20 49796469 Ki = 1400 nM T94033 C4MK5H 49796471 Ki > 21000 nM T94033 C75HOB 49796472 Ki = 11800 nM T94033 CS90ZF 49796473 Ki = 1600 nM T94033 C0OYG1 49796860 Ki = 10 nM T94033 C93ZMF 49796861 Ki = 150 nM T94033 CB2M0F 49796862 Ki = 2 nM T94033 CF9UQ8 49796863 Ki = 100 nM T94033 CGC5D9 49796864 Ki = 18 nM T94033 C01AHI 49796865 Ki = 1112 nM T94033 C6ZD3K 49796866 Ki = 18 nM T94033 CP04HB 49796867 Ki = 8 nM T94033 C5EMZ1 49796869 Ki = 235 nM T94033 CUOJ27 49796870 Ki = 550 nM T94033 C3VWR1 49796871 Ki = 16 nM T94033 CXUM36 49820499 Ki = 4100 nM T94033 CX7SA8 49820500 Ki = 5800 nM T94033 CS8FY6 49820655 Ki = 2343 nM T94033 C6OIW8 49820657 Ki = 3600 nM T94033 CL8UV3 49820969 Ki = 3125 nM T94033 C2B5EC 49820973 Ki = 1240 nM T94033 CU1DK9 49835415 Ki = 1 nM T94033 C0OQ8N 49835557 Ki = 0.39 nM T94033 CSB80A 49837842 Ki = 170000 nM T94033 C84XTM 49859969 Ki = 600 nM T94033 C78QKE 49864328 Ki > 25000 nM T94033 CFIW73 49864329 Ki > 25000 nM T94033 CDZ3B0 49864350 Ki > 25000 nM T94033 CLW9I6 49864373 Ki > 25000 nM T94033 CSZ3P1 49864435 Ki > 25000 nM T94033 CZR1W9 49864436 Ki > 25000 nM T94033 C5YH3T 49864437 Ki > 25000 nM T94033 CK5G4W 49864458 Ki > 25000 nM T94033 CLOY62 49864459 Ki > 25000 nM T94033 CR8JK9 49864483 Ki > 25000 nM T94033 CVDF05 50908868 IC50 = 10600 nM T94033 CCJ61A 51003503 Ki = 1.5 nM T94033 C9C1OQ 51003504 Ki = 1.1 nM T94033 CA3M0B 51003505 Ki = 3 nM T94033 C45UCD 51003506 Ki = 0.27 nM T94033 CD5K7M 51003507 Ki = 0.27 nM T94033 CZCO60 51035176 IC50 = 510 nM T94033 C1FL6J 52941173 IC50 = 67900 nM T94033 CQ91YB 53317095 Ki = 0.015 nM T94033 CNX09I 53317096 Ki = 8 nM T94033 C54GJP 53317109 Ki = 1.25 nM T94033 CA86OS 53317375 Ki = 1000000 nM T94033 CKP81R 53318397 Ki = 37 nM T94033 CKLQ81 53318398 Ki = 67 nM T94033 CY6V5L 53319728 Ki = 0.5 nM T94033 CQ4T1M 53319729 Ki = 34 nM T94033 CW6H9F 53320162 Ki = 2.9 nM T94033 C1RYX8 53320283 Ki = 1.7 nM T94033 CI5L4V 53320316 Ki = 0.68 nM T94033 CLU30N 53321021 Ki = 1.8 nM T94033 C7W2CT 53321022 Ki = 0.93 nM T94033 C4TWJ1 53321023 Ki = 1.6 nM T94033 CHQ59F 53321024 Ki = 50 nM T94033 CPFB49 53321025 Ki = 0.77 nM T94033 CLO86W 53321180 Ki = 860 nM T94033 CGZC91 53321290 Ki = 1000000 nM T94033 C7QEI1 53321291 Ki = 800000 nM T94033 C3RB9P 53322357 Ki = 1.3 nM T94033 CAD4I3 53322365 Ki = 2.3 nM T94033 CFOI53 53322612 Ki = 32000 nM T94033 CG1Z2U 53323724 Ki = 1.8 nM T94033 CJ8YU2 53323725 Ki = 1.8 nM T94033 C3LE1Q 53323726 Ki = 4.1 nM T94033 CWA7B3 53323948 Ki = 1000000 nM T94033 C5DJ9S 53324132 Ki = 9.6 nM T94033 C2K9VJ 53324991 Ki = 0.125 nM T94033 C1W9RD 53324992 Ki = 1.1 nM T94033 C85KEJ 53325003 Ki = 4.8 nM T94033 CP4S9V 53325004 Ki = 1.6 nM T94033 CO6TG4 53325236 Ki = 1000000 nM T94033 CO0R2M 53325237 Ki = 1000000 nM T94033 C3UPS7 53326281 Ki = 0.75 nM T94033 CE9VT8 53326282 Ki = 1.6 nM T94033 C2QGK5 53326293 Ki = 1.5 nM T94033 CJ5X6M 53326294 Ki = 3.5 nM T94033 C36ABV 53326295 Ki = 0.73 nM T94033 C57RVG 53326296 Ki = 7 nM T94033 CH59WQ 53326297 Ki = 85 nM T94033 C50NGR 53326298 Ki = 0.93 nM T94033 CWHX59 53326648 Ki = 2 nM T94033 CA6GQ5 53341037 Ki > 11500 nM T94033 CIKQ81 53345652 Ki > 130 nM T94033 CXWS90 53345968 Ki > 1000 nM T94033 CCR6H5 53357861 IC50 = 14000 nM T94033 CI9GP5 53357862 IC50 = 5100 nM T94033 C52ZET 53357863 IC50 = 7800 nM T94033 C53JUT 53357864 IC50 = 6700 nM T94033 C9YK0S 53357865 IC50 = 5200 nM T94033 CB08CW 53379392 Ki = 5.2 nM T94033 C6XNM0 53380822 Ki = 430 nM T94033 C1KFQ0 53380823 Ki = 950 nM T94033 C7JWD0 53380936 Ki = 690 nM T94033 C97KGD 53380937 Ki = 800 nM T94033 CKV6Q2 53380938 Ki = 310 nM T94033 C47WIH 53380939 Ki = 480 nM T94033 CY3RO0 53380940 Ki = 330 nM T94033 C3R8PW 53380941 Ki = 290 nM T94033 C7O2RL 53391543 IC50 = 758577.58 nM T94033 CW01RN 53391545 IC50 = 363078.05 nM T94033 C4LA2P 53391547 IC50 = 89000 nM T94033 CM5L4F 53391856 IC50 > 2500000 nM T94033 C4X2PJ 53391857 IC50 > 3000000 nM T94033 C3N9LW 53391859 IC50 > 3000000 nM T94033 CN03KJ 53391966 IC50 > 2000000 nM T94033 CJ8EA2 53391968 IC50 = 19952623.15 nM T94033 CQ67BZ 53391970 IC50 = 12589254.12 nM T94033 CX5EV0 53391972 IC50 > 16000000 nM T94033 CYP10E 53391974 IC50 > 25000000 nM T94033 CP45DY 53391976 IC50 = 501187.23 nM T94033 CR8XO9 53391978 IC50 > 3000000 nM T94033 C92UBT 53392081 IC50 > 2000000 nM T94033 C4HB3V 53392251 IC50 = 5500 nM T94033 CKY2V1 53392252 IC50 = 37000 nM T94033 CW2T7R 53392254 IC50 = 7244.36 nM T94033 CL7D1H 53392255 IC50 = 375000 nM T94033 CLGU52 53392340 IC50 = 121000 nM T94033 CH1QR8 53392341 IC50 = 30000 nM T94033 CXE2T1 53392969 IC50 > 7000000 nM T94033 C2RZD4 53392971 IC50 = 129000 nM T94033 CAS01X 53392973 IC50 > 7100000 nM T94033 CT62JM 53392975 IC50 = 371535.23 nM T94033 C4V2OJ 53483931 Ki = 1710 nM T94033 CD0YA3 53484213 Ki = 880 nM T94033 C7DV0R 53484214 Ki = 1970 nM T94033 C3KCW1 53484215 Ki = 1750 nM T94033 CJ12OY 53484216 Ki = 2270 nM T94033 CV60BK 53488415 Ki = 3280 nM T94033 CGP67H 53706682 Ki = 32400 nM T94033 C8SCH2 53800364 IC50 = 180000 nM T94033 C9GFU3 53864431 IC50 = 55000 nM T94033 C16KAQ 53954748 IC50 = 95000 nM T94033 CK7V4P 54039220 Ki = 651 nM T94033 CBJQ98 54132077 IC50 = 53170 nM T94033 CHB03N 54252937 Ki > 4000 nM T94033 CEIQ26 54352954 IC50 > 100000 nM T94033 CQNW76 54507330 IC50 = 75000 nM T94033 C2FS3H 54555233 IC50 = 400000 nM T94033 CP6I2C 54585528 IC50 > 133000 nM T94033 CDF47K 54587541 IC50 = 150000 nM T94033 C9I4OP 54738720 Ki > 5000 nM T94033 CPGD29 56598201 IC50 > 50000 nM T94033 C6QCK2 56598333 IC50 > 50000 nM T94033 C17MSO 56640092 Ki = 45.4 nM T94033 CGP7Y6 56640160 Ki = 7.2 nM T94033 C30AJK 56640226 Ki = 510 nM T94033 C8U4OD 56649692 IC50 > 1000000 nM T94033 C1U2ZB 56655960 IC50 = 1030 nM T94033 CGW36Z 56655962 IC50 = 2500 nM T94033 CG40BF 56656038 IC50 = 450 nM T94033 CH76DQ 56659112 Ki = 0.005 nM T94033 C9YXM2 56659587 IC50 > 1340000 nM T94033 CA32CM 56659850 Ki = 74 nM T94033 C6OI5V 56660094 Ki = 660 nM T94033 CKFI81 56660095 Ki = 350 nM T94033 C8O0CK 56661932 Ki = 4600 nM T94033 CKO4M6 56663319 Ki = 68 nM T94033 C9XCR1 56665418 Ki = 5430 nM T94033 C74FZH 56665419 Ki = 5200 nM T94033 C2T1WM 56665604 IC50 = 19300 nM T94033 CMG9H6 56666511 IC50 > 580000 nM T94033 CS9PL8 56669578 IC50 > 2000000 nM T94033 CCM80T 56670171 Ki = 6.7 nM T94033 C0M3AE 56673432 IC50 > 1480000 nM T94033 CI6RX7 56673433 IC50 > 590000 nM T94033 C8ESB6 56673691 Ki = 1.29 nM T94033 CXGO13 56673692 Ki = 0.891 nM T94033 CGM2J4 56673694 Ki = 66 nM T94033 C4T6NO 56673695 Ki = 1610 nM T94033 CL35DR 56675717 Ki = 62500 nM T94033 C7DE8I 56676739 IC50 > 1340000 nM T94033 CE4AT6 56676740 IC50 > 400000 nM T94033 C8CN9W 56676741 IC50 = 560000 nM T94033 C1TH3W 56677006 Ki = 13.5 nM T94033 CY34VE 56677007 Ki = 29 nM T94033 C7Z6GI 56679017 Ki = 13700 nM T94033 CN2H9U 56679018 Ki = 8910 nM T94033 C6PIH2 56679020 Ki = 6890 nM T94033 C5LVJ2 56680051 IC50 > 640000 nM T94033 CKF2M0 56680052 IC50 > 650000 nM T94033 C72IHP 56680339 Ki = 9.8 nM T94033 C1ZLR5 56682336 Ki = 39200 nM T94033 CT7U8L 56683905 Ki = 300 nM T94033 C3CDB4 56683906 Ki = 370 nM T94033 CXTP34 56947156 Ki = 3.7 nM T94033 CS8A2N 56947157 Ki = 5.2 nM T94033 C9MW7H 56947159 Ki = 0.63 nM T94033 C0RP5S 56947160 Ki = 2.2 nM T94033 C0QEJ6 56947161 Ki = 0.798 nM T94033 C8UHN3 56949979 IC50 > 100000 nM T94033 C2K8UT 56950928 Ki = 23400 nM T94033 CH1EI8 56954620 Ki = 2020 nM T94033 C4EHU8 56954732 Ki = 6520 nM T94033 C5C8XO 56954733 Ki = 3517 nM T94033 CST4F0 56954834 Ki = 26.8 nM T94033 CRK92A 56954952 Ki = 6175 nM T94033 CA0G3M 57133681 Ki = 230000 nM T94033 CN6CZ8 57154289 IC50 > 500000 nM T94033 CLU95A 57325502 IC50 > 62000 nM T94033 CV42AN 57390824 IC50 > 62000 nM T94033 C1GIV7 57390825 IC50 > 62000 nM T94033 CM7FT5 57390879 IC50 > 125000 nM T94033 CB57DW 57391171 Ki = 670 nM T94033 CWJ4I7 57391565 Ki = 5000 nM T94033 CPBW48 57392333 Ki = 330000 nM T94033 C7APO2 57392934 Ki = 330 nM T94033 CZ2A0S 57392935 Ki = 28 nM T94033 CP4MW8 57393205 Ki = 132700 nM T94033 CX16KB 57393324 Ki = 200 nM T94033 CXV4U9 57394359 IC50 > 62000 nM T94033 C6EWL9 57394677 Ki = 240 nM T94033 CQ9V5U 57394920 Ki = 19580 nM T94033 C8T2ZJ 57395044 Ki = 18 nM T94033 CL2JE5 57395841 Ki = 680000 nM T94033 CZ6FM4 57395852 IC50 = 9800 nM T94033 CNH2M8 57397633 IC50 = 98000 nM T94033 C1KMO0 57397634 IC50 = 73000 nM T94033 CIC2U6 57397927 IC50 > 62000 nM T94033 C9F4OL 57398232 Ki = 750 nM T94033 C5OAB7 57398233 Ki = 23 nM T94033 CY39KP 57398234 Ki = 19 nM T94033 CA1F6J 57399306 IC50 = 26200 nM T94033 CODX48 57399879 Ki = 1700 nM T94033 C93VSX 57399880 Ki = 240 nM T94033 C5WOZ3 57399881 Ki = 290 nM T94033 C9ZL5X 57400230 Ki = 150 nM T94033 CPZR79 57400272 Ki = 320 nM T94033 C0IGQ9 57400533 IC50 = 110 nM T94033 CKV6R8 57401327 IC50 > 62000 nM T94033 CS2ZY1 57401658 Ki = 2000 nM T94033 CES6D2 57403083 IC50 > 62000 nM T94033 CG90KP 57403382 Ki = 260 nM T94033 C3CKA6 57403383 Ki = 810 nM T94033 C4OB6Z 57403384 Ki = 3000 nM T94033 CKI4S8 57403776 Ki = 760 nM T94033 C5MX2D 57404340 IC50 > 50000 nM T94033 CL1T6Z 57411954 Ki = 0.259 nM T94033 C4R2LU 57594784 IC50 > 100000 nM T94033 C63FQC 57803696 Ki = 570 nM T94033 CLV91D 57803729 Ki = 4470 nM T94033 CEH39Z 57803776 Ki = 1190 nM T94033 C2W7GY 57803799 Ki = 790 nM T94033 CU4N3X 57803861 Ki = 710 nM T94033 CEG27C 57803875 Ki = 750 nM T94033 CI6U8B 57803906 Ki = 1200 nM T94033 C6X3ER 57803948 Ki = 640 nM T94033 CH2QT8 57804013 Ki = 1670 nM T94033 C45OXB 57804023 Ki = 190 nM T94033 CFMO72 57804069 Ki = 760 nM T94033 CTE30K 57842560 Ki > 13000 nM T94033 C0C6UB 57842624 Ki = 4000 nM T94033 C7XY5A 57842673 Ki > 13000 nM T94033 CU9S6K 57842710 Ki > 13000 nM T94033 CL8T7M 57842742 Ki > 13000 nM T94033 C41NSR 57842812 Ki = 180 nM T94033 C9XW1C 57842830 Ki > 10000 nM T94033 CWF0C3 57842850 Ki = 5800 nM T94033 C73CPB 57842913 Ki = 6700 nM T94033 CB5F0H 57942680 Ki = 5700 nM T94033 C8GXF1 57942687 Ki = 3400 nM T94033 CO52PA 57942693 Ki = 6700 nM T94033 CS23DW 57942743 Ki = 4400 nM T94033 C0DO5P 57942817 Ki = 4400 nM T94033 CV0KZ6 57942834 Ki = 4900 nM T94033 C0KRC1 57942835 Ki = 6400 nM T94033 C60HCV 57976401 Ki > 11500 nM T94033 CHB27Y 57976410 Ki > 13340 nM T94033 CM8UJ7 57976444 Ki > 13000 nM T94033 CQ71KE 57976446 Ki > 15000 nM T94033 CXL75F 58630486 Ki > 15000 nM T94033 C3OA5C 58789089 Ki = 2400 nM T94033 C2W1UT 58789135 Ki = 2900 nM T94033 CT9C1Z 58789193 Ki = 2800 nM T94033 COPW56 58834156 Ki = 140 nM T94033 CSC0L5 59020200 Ki = 2578 nM T94033 C91APY 59095797 IC50 > 33000 nM T94033 C69SED 59095888 IC50 > 33000 nM T94033 CPW2H7 59315536 Ki > 10000 nM T94033 CO38AC 59402011 Ki > 13000 nM T94033 CMU38J 59432238 IC50 > 100000 nM T94033 C7IO5P 60150643 Ki = 1.1 nM T94033 CE5A7B 60162406 Ki = 13870 nM T94033 CWCA65 66573845 IC50 > 500000 nM T94033 CWOD93 66744646 Ki > 11500 nM T94033 CSAQ19 66818162 Ki = 2500 nM T94033 CG9UM3 66818450 Ki = 1285 nM T94033 CG0TZ3 66818504 Ki = 4850 nM T94033 CU6E0A 66818541 Ki = 2216 nM T94033 C89BXR 66818555 Ki = 2100 nM T94033 C6LD2R 66818559 Ki = 2808 nM T94033 C6CP8D 66818568 Ki = 2677 nM T94033 CKD8I1 66818569 Ki = 2105 nM T94033 C05LHZ 66818575 Ki = 1636 nM T94033 C9LTK3 66818589 Ki = 3400 nM T94033 C9GM3F 66818639 Ki = 3973 nM T94033 C4U7SZ 66818677 Ki = 2530 nM T94033 CL8D0V 66818717 Ki = 4202 nM T94033 C41RKZ 66818743 Ki > 2500 nM T94033 C6Q8FO 66818744 Ki = 2406 nM T94033 CE53KG 66818763 Ki = 2816 nM T94033 CJA30C 66818765 Ki = 1785 nM T94033 C5LU1Z 66818766 Ki = 2467 nM T94033 CP18VA 66818813 Ki = 744 nM T94033 CF4PT6 66818819 Ki = 3540 nM T94033 CYB76J 66818882 Ki = 3250 nM T94033 CRH5O7 66818889 Ki > 2500 nM T94033 CGI6B3 66819113 Ki = 2680 nM T94033 C4JV1L 66820910 Ki = 1562 nM T94033 C62LDA 66821311 Ki = 4061 nM T94033 CE6JP2 66911194 IC50 = 17 nM T94033 CGH09I 66911211 IC50 = 126 nM T94033 CKWQ82 67155200 Ki = 8 nM T94033 CY05ND 67155277 IC50 = 890 nM T94033 CA0GE1 67155403 IC50 = 23 nM T94033 CN51PD 67155431 IC50 = 31 nM T94033 C0SDB3 68020667 Ki = 14143 nM T94033 C17JAZ 68284084 IC50 > 30000 nM T94033 CE79VS 68440006 Ki = 3600 nM T94033 CK59IZ 68788696 Ki = 1056 nM T94033 CGA3T2 68789018 Ki = 1289 nM T94033 CC0J3V 68790735 Ki = 1642 nM T94033 CA5DG8 69249482 Ki = 1800 nM T94033 CQY32W 69295008 Ki = 6900 nM T94033 CA49UK 69520512 Ki = 0.5 nM T94033 C0KB4O 69641445 Ki = 11000 nM T94033 CO3Z8Y 69654811 Ki = 220 nM T94033 C7BF4M 69953169 Ki = 310 nM T94033 CO5AI8 70004055 Ki = 1.1 nM T94033 C6AU1R 70252985 Ki > 13300 nM T94033 CTO5I6 70253788 Ki > 13300 nM T94033 C8A7ZJ 70306716 Ki = 1700 nM T94033 C0WKD9 70662368 IC50 = 4000 nM T94033 CUOA08 70681485 Ki = 0.004 nM T94033 C4IFW3 70683249 Ki = 667 nM T94033 C28CEG 70685001 IC50 > 10000 nM T94033 CND19T 70685163 IC50 = 130 nM T94033 CJY20L 70686249 Ki = 481000 nM T94033 C0M1ND 70687125 Ki = 19 nM T94033 C7U9OA 70687171 IC50 > 10000 nM T94033 CN38UY 70687492 Ki = 137 nM T94033 CFJ80W 70690392 Ki = 2731000 nM T94033 C2N8MX 70697537 Ki = 240 nM T94033 C9EL3C 71260387 Ki > 13300 nM T94033 CV3M4L 71449633 Ki = 250000 nM T94033 CXT97V 71449635 Ki = 175000 nM T94033 C45SHM 71451304 Ki > 20000 nM T94033 C28YUT 71451445 Ki = 160000 nM T94033 CWQ5O0 71451447 Ki = 187000 nM T94033 C1NKU9 71452612 Ki = 18 nM T94033 C30XPC 71453256 IC50 > 500000 nM T94033 CGM4Q1 71453258 Ki = 223000 nM T94033 C5ZL0G 71453261 IC50 > 500000 nM T94033 C39ZJF 71453263 Ki = 15600 nM T94033 CV3T2M 71453265 Ki = 83000 nM T94033 C5JKU3 71454986 Ki = 165000 nM T94033 C2H9WA 71454988 Ki = 32000 nM T94033 CET86A 71454990 Ki = 28000 nM T94033 C0XV2L 71455698 IC50 = 100000 nM T94033 CQIB21 71456772 IC50 > 500000 nM T94033 CHNV94 71456774 Ki = 71000 nM T94033 C3MT0E 71456776 Ki = 245000 nM T94033 CP3AQ0 71457928 Ki = 178 nM T94033 C1UOK5 71458276 EC50 = 7500 nM T94033 CXB02M 71458628 IC50 > 500000 nM T94033 CK7DL1 71458630 Ki = 120000 nM T94033 CPJG15 71458632 Ki = 165000 nM T94033 C51OSR 71458634 IC50 > 500000 nM T94033 CX37BW 71458636 Ki = 172000 nM T94033 C04EON 71458638 Ki = 12300 nM T94033 CPDA60 71460459 IC50 > 500000 nM T94033 CAK34J 71461597 IC50 = 500 nM T94033 CC4P2V 71462161 IC50 > 500000 nM T94033 CU8WH5 71462163 IC50 > 500000 nM T94033 CK90PE 71462165 Ki = 60000 nM T94033 CEXT02 71475974 Ki = 10700 nM T94033 C9TE8A 71475975 Ki = 2400 nM T94033 CI6FA7 71475976 Ki = 11200 nM T94033 C6E1GM 71475977 Ki = 530 nM T94033 CLE0Y3 71476908 Ki = 18000 nM T94033 CAJ0C4 71476909 Ki = 4000 nM T94033 C5KQ9M 71476910 Ki = 7600 nM T94033 CUBF31 71477064 Ki = 13000 nM T94033 CRD18E 71477065 Ki = 10600 nM T94033 CHC7K2 71477066 Ki = 8530 nM T94033 CZH38E 71477067 Ki = 5820 nM T94033 CQT08V 71477068 Ki = 85000 nM T94033 C24WTK 71477222 Ki = 64000 nM T94033 C1E0MZ 71477223 Ki = 174000 nM T94033 C6CBP2 71477224 Ki = 100000 nM T94033 CR47VE 71477225 Ki = 103000 nM T94033 CEA26W 71477226 Ki = 115000 nM T94033 CSXC62 71477380 Ki = 13800 nM T94033 CE3LD8 71477381 Ki = 7400 nM T94033 CF67HS 71477382 Ki = 63000 nM T94033 CAOD57 71477383 Ki = 13000 nM T94033 CP7TO4 71477384 Ki = 15000 nM T94033 CT16CB 71477529 Ki = 30000 nM T94033 CUC56G 71477530 IC50 > 500000 nM T94033 CN7IV2 71477531 IC50 > 500000 nM T94033 CQ7RZ1 71477532 IC50 > 500000 nM T94033 C4HPE8 71477533 IC50 > 500000 nM T94033 CIU9J6 71477683 Ki = 66000 nM T94033 C3EOG6 71477684 Ki = 201000 nM T94033 C5GKW9 71477685 Ki = 52000 nM T94033 CH3AO9 71477686 Ki = 37000 nM T94033 C5C4IM 71477687 Ki = 29000 nM T94033 CI5U2V 71477829 Ki = 88000 nM T94033 C2WGZ0 71477830 Ki = 30000 nM T94033 C15WQM 71477831 Ki = 75000 nM T94033 CD8X3F 71477832 Ki = 125000 nM T94033 CSB35T 71477833 Ki = 10600 nM T94033 C1N4FS 71477979 Ki = 7400 nM T94033 C0H8NK 71477980 Ki = 17000 nM T94033 CPHV01 71477981 Ki = 8200 nM T94033 C6X5KL 71477982 Ki = 5100 nM T94033 C45FPN 71478120 Ki = 16500 nM T94033 CU2VL3 71478121 Ki = 6000 nM T94033 C4OGP2 71478122 Ki = 32000 nM T94033 C4IXP0 71478123 Ki = 930 nM T94033 CBQU35 71517738 IC50 = 65900 nM T94033 CPAL73 71517739 IC50 = 743000 nM T94033 CK0I1X 71533477 IC50 = 286000 nM T94033 CJPF90 71548883 Ki > 13000 nM T94033 C30ZKJ 71561420 Ki = 26420 nM T94033 CH32TL 71561557 Ki = 884 nM T94033 C83ZNH 71562308 IC50 = 1219 ug.mL-1 T94033 C8RW7E 71562631 Ki = 227 nM T94033 C4UHB2 71562760 Ki = 604 nM T94033 C0EM6D 71562761 Ki = 3250 nM T94033 CNS21T 71562882 Ki = 376 nM T94033 C3SBE2 71562883 Ki = 11210 nM T94033 C2NY0B 71563006 Ki = 12082 nM T94033 CG46AZ 71563007 Ki = 8510 nM T94033 C2O4SB 71563124 Ki = 5870 nM T94033 C4CT8O 71563125 Ki = 2950 nM T94033 C6I9DJ 71567884 Ki = 220 nM T94033 CC7Z0N 71567885 Ki = 36 nM T94033 C40CRP 71567886 Ki = 110 nM T94033 CG8X1C 71567887 Ki = 78 nM T94033 C5DU6Q 71568014 Ki > 15000 nM T94033 C4ICT8 71568015 Ki > 15000 nM T94033 C9BSO1 71568137 Ki = 32 nM T94033 C9TBN3 71568263 Ki = 1800 nM T94033 CXYQ68 71568403 Ki = 2100 nM T94033 C53BYN 71580813 Ki = 35 nM T94033 C57PCL 71580892 Ki = 330 nM T94033 CG1V9P 71627416 Ki > 13000 nM T94033 C9J7NH 71652207 Ki = 266 nM T94033 CLH52G 71654374 Ki = 1650 nM T94033 C8GDV7 71654376 Ki = 436 nM T94033 CY29LR 71654530 Ki = 675 nM T94033 C3K6PT 71654532 Ki = 77.8 nM T94033 C3X7FP 71654534 Ki = 5180 nM T94033 CCGP56 71654535 Ki = 1670 nM T94033 CZG3Y9 71654536 Ki = 2690 nM T94033 C62ZTJ 71660643 IC50 > 33000 nM T94033 C5D2OL 71698598 Ki > 100000 nM T94033 CGYN76 71698686 Ki > 100000 nM T94033 CD0Z5K 71698687 Ki > 100000 nM T94033 C0DUT2 71698688 Ki > 100000 nM T94033 C60JTA 71698689 Ki > 100000 nM T94033 C35ZJV 71698690 Ki > 100000 nM T94033 C9XSB5 71698770 Ki > 100000 nM T94033 CRN95M 71698771 Ki > 100000 nM T94033 C0LW4G 71698774 Ki > 100000 nM T94033 CH26JR 71698775 Ki > 100000 nM T94033 C0WR9F 71699124 Ki > 100000 nM T94033 CZKL39 71699125 Ki > 100000 nM T94033 C27TZK 71699126 Ki > 100000 nM T94033 CD12FS 71699127 Ki > 100000 nM T94033 CFN7Q4 71699199 Ki > 100000 nM T94033 C7RTF0 71699200 Ki > 100000 nM T94033 C8JE0W 71699201 Ki = 53000 nM T94033 CRAG19 71699203 Ki > 100000 nM T94033 CYAH23 71699286 Ki > 100000 nM T94033 CM8E7F 71699287 Ki > 100000 nM T94033 C9Y3DN 71699288 Ki > 100000 nM T94033 CD53RA 71716975 Ki > 120000 nM T94033 CSP5T2 71716976 Ki > 120000 nM T94033 CU09NX 71717260 IC50 = 3900 nM T94033 CQ3K2V 71719191 Ki = 8017 nM T94033 C08BOY 71734677 IC50 = 260 nM T94033 C4TP1M 71748092 Ki = 7.3 nM T94033 CVM7Y6 71748093 Ki = 63 nM T94033 C8HZ6Q 71748094 Ki = 34 nM T94033 C6CB0G 71748095 Ki = 32 nM T94033 C2Z7XJ 71748113 Ki = 52 nM T94033 C5B4MS 71748117 Ki = 78 nM T94033 C5RSD4 71818404 IC50 = 640 nM T94033 CVPL10 71818549 IC50 = 1900 nM T94033 CVCM38 71818688 IC50 = 830 nM T94033 CA56TS 71818689 IC50 = 1100 nM T94033 CK2XH0 71818692 IC50 = 480 nM T94033 CXV8Z4 71818829 IC50 = 82 nM T94033 C7UY4N 71818830 IC50 = 370 nM T94033 C6X2FC 71818831 IC50 = 310 nM T94033 C80YBP 71818832 IC50 = 39 nM T94033 CXV20J 71818964 IC50 = 160 nM T94033 CM83VP 72163524 IC50 > 10000 nM T94033 CRBH34 72164200 IC50 > 33000 nM T94033 CWNZ45 72164201 IC50 > 33000 nM T94033 CBVO02 72164443 Ki > 13000 nM T94033 C1W9NH 72164444 Ki > 13000 nM T94033 C6Z3IC 72164445 Ki = 10300 nM T94033 C0CGB5 72164564 Ki > 13000 nM T94033 CN37EY 72164565 Ki > 13000 nM T94033 CIT3O5 72164566 Ki > 13000 nM T94033 C80OFE 72164567 Ki > 13000 nM T94033 CD01PR 72164568 Ki = 9400 nM T94033 C85RCG 72164697 Ki > 13000 nM T94033 CP4M2G 72164698 Ki > 13000 nM T94033 C0EWD8 72164699 Ki = 9400 nM T94033 C9G4PK 72200999 IC50 = 10.5 nM T94033 CG8Z7P 72206621 IC50 = 7 nM T94033 CK34ZH 72550138 Ki > 10000 nM T94033 CT45ER 72550807 Ki > 10000 nM T94033 C46TNC 72550811 Ki > 10000 nM T94033 CXM6C2 72550813 Ki > 13300 nM T94033 CLI36U 72551247 Ki = 11000 nM T94033 C97DUL 72708122 IC50 > 100000 nM T94033 CW3QR2 72712049 Ki = 14 nM T94033 CAL2W7 72712050 Ki = 16 nM T94033 C2A4TH 72712051 Ki = 90 nM T94033 CN73TI 72712053 Ki = 31 nM T94033 C3J8RV 72712070 Ki = 755 nM T94033 CM1OK7 72792543 IC50 = 230 nM T94033 CBP05V 72792607 IC50 = 1300 nM T94033 CYXT24 72792608 IC50 = 13 nM T94033 CO89NF 72792609 IC50 = 13 nM T94033 CC50RS 72792610 IC50 = 20 nM T94033 CCEZ71 72792672 IC50 = 10 nM T94033 CFRI96 72792673 IC50 = 27 nM T94033 C86RTS 72792674 IC50 = 20 nM T94033 CI5U3J 72792675 IC50 = 72 nM T94033 CQ08NT 72792744 IC50 = 80 nM T94033 CWB62R 72792745 IC50 = 1813 nM T94033 CA8WG3 72792746 IC50 = 41 nM T94033 CR17NL 72792747 IC50 = 65 nM T94033 C1MBU7 72793747 IC50 > 50000 nM T94033 C6BY5D 72793776 IC50 > 50000 nM T94033 C1DI8A 72793778 IC50 = 8400 nM T94033 C9TOS3 73345471 Ki = 0.37 nM T94033 CF07MV 73345564 Ki = 260 nM T94033 C7KJ5L 73345607 Ki = 6.7 nM T94033 CW84BZ 73345684 IC50 > 100000 nM T94033 CT21AC 73345685 IC50 > 100000 nM T94033 CPF63K 73345705 IC50 = 1141000 nM T94033 C84SCY 73345706 IC50 = 6400 nM T94033 CSQ7U6 73345707 IC50 = 257000 nM T94033 C5W8JA 73345708 IC50 = 20000 nM T94033 C5HWZ3 73345709 IC50 = 46000 nM T94033 CQE45K 73345710 IC50 = 54000 nM T94033 CR34QD 73345711 IC50 = 46000 nM T94033 C7BG9I 73345713 IC50 = 672000 nM T94033 C8O3PT 73345716 IC50 = 106000 nM T94033 CFC2Y6 73345717 IC50 = 507000 nM T94033 C4FQ0W 73345765 Ki = 11 nM T94033 CCD54H 73345766 Ki = 1.8 nM T94033 CO4A1M 73345767 Ki = 1700 nM T94033 CC2FW1 73345771 Ki = 85 nM T94033 CNH82E 73346602 Ki = 0.36 nM T94033 CN4RC6 73346747 Ki = 0.2 nM T94033 CRK20G 73346850 Ki = 3 nM T94033 CE20RU 73347003 Ki = 0.56 nM T94033 CDQP51 73347119 Ki > 50000 nM T94033 C5YH0Z 73347129 Ki = 1.3 nM T94033 C3JN8A 73347180 IC50 > 500000 nM T94033 CQ7PY1 73347205 IC50 = 21000 nM T94033 C8JZN2 73347206 IC50 = 126000 nM T94033 C7JAE5 73347207 IC50 = 821000 nM T94033 C50JPH 73347208 IC50 = 2776000 nM T94033 C7AD5S 73347209 IC50 = 507000 nM T94033 CHJF63 73347210 IC50 = 13000 nM T94033 C5NLQ1 73347211 IC50 = 68000 nM T94033 C9G1UX 73347212 IC50 = 15000 nM T94033 C0KPO1 73347215 IC50 = 17000 nM T94033 C98IGZ 73347216 IC50 = 183000 nM T94033 C5QTF3 73347217 IC50 = 3326000 nM T94033 CZ4ET2 73347356 Ki = 10 nM T94033 C5AMR2 73348056 IC50 < 1000 nM T94033 CH49DP 73348103 Ki = 0.8 nM T94033 C8HJ5Y 73348104 Ki = 5.6 nM T94033 CQ8Y3U 73348105 Ki = 0.22 nM T94033 CVE63C 73348106 Ki = 0.19 nM T94033 C28YDF 73348107 Ki = 0.27 nM T94033 CWG97H 73348174 Ki = 0.46 nM T94033 C7HWF2 73348631 Ki = 0.6 nM T94033 CG2YC8 73348714 IC50 = 1713000 nM T94033 CKJ4Z5 73348715 IC50 = 137000 nM T94033 CHV4R9 73348716 IC50 = 300000 nM T94033 C0KZM9 73348717 IC50 = 298000 nM T94033 CT0K2N 73348718 IC50 = 318000 nM T94033 CH25NM 73348720 IC50 = 422000 nM T94033 C5SR4V 73348721 IC50 = 42000 nM T94033 C7CX3N 73348722 IC50 = 168000 nM T94033 C09PTB 73348723 IC50 = 680000 nM T94033 CGI64K 73348724 IC50 = 26000 nM T94033 C8F7OD 73348725 IC50 = 2803000 nM T94033 C8Z6MJ 73348726 IC50 = 2989000 nM T94033 C6AV2Y 73348727 IC50 = 29000 nM T94033 CT0ZK7 73348728 IC50 = 593000 nM T94033 C5SM8A 73348729 IC50 = 3386000 nM T94033 CQF46R 73348759 Ki = 210 nM T94033 CJG30R 73348764 Ki = 85 nM T94033 CUD26E 73348765 Ki = 8.6 nM T94033 CST16Q 73348766 Ki = 350 nM T94033 CSQ41U 73348767 Ki = 5.5 nM T94033 C7Y3ZB 73348933 Ki = 16600 nM T94033 CP62UY 73349650 Ki = 0.43 nM T94033 C7IZ4U 73349651 Ki = 0.58 nM T94033 CHL60U 73349652 Ki = 0.85 nM T94033 CAJ7O5 73350148 Ki > 1000000 nM T94033 CM3PH8 73350210 Ki > 50000 nM T94033 CYL2K9 73350270 IC50 = 5000 nM T94033 C1EPR4 73350271 IC50 = 170000 nM T94033 CBM59R 73350292 IC50 = 2206000 nM T94033 C20AJY 73350293 IC50 = 7000 nM T94033 C9IU2M 73350294 IC50 = 3542000 nM T94033 C8XLN3 73350295 IC50 = 1887000 nM T94033 C7IHX6 73350296 IC50 = 2545000 nM T94033 CTA7Z8 73350297 IC50 = 5800 nM T94033 C7HA2V 73350298 IC50 = 394000 nM T94033 CQI6Z7 73350300 IC50 = 262000 nM T94033 CIX40D 73350301 IC50 = 341000 nM T94033 CHF47P 73350338 Ki = 41 nM T94033 C5VP6W 73350339 Ki = 73 nM T94033 CK45HD 73350340 Ki = 0.8 nM T94033 C60BNQ 73350342 Ki = 2.6 nM T94033 C1GKO4 73350343 Ki > 42 nM T94033 CSI16A 73350344 Ki = 36 nM T94033 CL8EG7 73350757 Ki = 0.02 nM T94033 CSN9V7 73351187 Ki = 0.42 nM T94033 CJED29 73351188 Ki = 0.45 nM T94033 COIS05 73351606 Ki = 0.3 nM T94033 C4LIK9 73351716 Ki = 2 nM T94033 C36EPY 73351772 IC50 > 500000 nM T94033 COBX03 73351777 IC50 = 79000 nM T94033 CSN8Q5 73351800 IC50 = 2576000 nM T94033 CS5TM0 73351801 IC50 = 69000 nM T94033 CT2YE6 73351802 IC50 = 2956000 nM T94033 CNQ15I 73351803 IC50 = 2164000 nM T94033 C49YPV 73351804 IC50 = 446000 nM T94033 CE29FZ 73351805 IC50 = 82000 nM T94033 C7QX3G 73351806 IC50 = 2710000 nM T94033 CAI8Y4 73351809 IC50 = 2328000 nM T94033 CV4T2U 73351810 IC50 = 2462000 nM T94033 C2NEV3 73351853 Ki = 84 nM T94033 CNFV61 73351854 Ki = 31 nM T94033 CO0I9J 73351855 Ki = 173 nM T94033 CX1WJ7 73351856 Ki = 8.7 nM T94033 C4CD7U 73351857 Ki = 150 nM T94033 CF12CM 73351860 Ki = 33 nM T94033 CQD32M 73352663 Ki = 0.78 nM T94033 C9IDO7 73352664 Ki = 0.32 nM T94033 CX75KM 73352665 Ki = 1.8 nM T94033 CY2JB6 73352666 Ki < 0.1 nM T94033 CAD90P 73352667 Ki = 0.19 nM T94033 C3X9VM 73352762 Ki = 0.24 nM T94033 C60JSR 73353029 Ki = 720000 nM T94033 CW4Z7M 73353192 Ki = 4.6 nM T94033 CKA2H6 73353276 IC50 = 200000 nM T94033 CN82CP 73353277 IC50 = 11000 nM T94033 C0OVW8 73353279 IC50 = 1262000 nM T94033 CB1M2Q 73353280 IC50 = 711000 nM T94033 C7MC1K 73353281 IC50 = 3013000 nM T94033 C4ZKC1 73353282 IC50 = 273000 nM T94033 C5SHZ4 73353283 IC50 = 582000 nM T94033 COI78M 73353284 IC50 = 44000 nM T94033 CZP8Y7 73353285 IC50 = 43000 nM T94033 CE71LX 73353286 IC50 = 294000 nM T94033 C69BHN 73353326 Ki = 160 nM T94033 C26QPS 73353327 Ki = 150 nM T94033 C7DGZ9 73353328 Ki = 65 nM T94033 CA2P1B 73353330 Ki = 33 nM T94033 C4J0AV 73354166 Ki = 0.5 nM T94033 C0B4DE 73354167 Ki = 0.23 nM T94033 CPQ9B4 73354563 Ki = 0.14 nM T94033 CPS6J3 73354766 IC50 = 88000 nM T94033 CLEH87 73354789 IC50 = 446000 nM T94033 C64RYQ 73354790 IC50 = 27000 nM T94033 C5CEX2 73354791 IC50 = 2873000 nM T94033 C2LRD4 73354792 IC50 = 31000 nM T94033 CJV4P0 73354793 IC50 = 13000 nM T94033 C0C3DO 73354794 IC50 = 378000 nM T94033 C0RQT9 73354795 IC50 = 458000 nM T94033 C09ZCK 73354796 IC50 = 2630000 nM T94033 C5TVR8 73354799 IC50 = 169000 nM T94033 CI83LO 73354800 IC50 = 3383000 nM T94033 C47KME 73354801 IC50 = 3153000 nM T94033 C8BX9N 73354802 IC50 = 54000 nM T94033 C3T2EK 73354803 IC50 = 9000 nM T94033 CUML80 73354804 IC50 = 194000 nM T94033 CNRW95 73354848 Ki = 4.6 nM T94033 COF2K0 73354849 Ki = 230 nM T94033 C3VFD6 73354850 Ki = 33 nM T94033 CL34CV 73354863 Ki = 3.5 nM T94033 C1U4BK 73355708 Ki = 0.5 nM T94033 C15ZAK 73355709 Ki = 0.09 nM T94033 CQI9X3 73355710 Ki = 0.16 nM T94033 C5U9CI 73355715 Ki = 0.0015 nM T94033 CDUR49 73356130 Ki = 300 nM T94033 CZ5LD9 73356131 Ki = 3.8 nM T94033 CXG0B8 73356296 IC50 > 10000 nM T94033 C37BVC 73356324 IC50 = 195000 nM T94033 CGD1T7 73356325 IC50 = 2430000 nM T94033 C93CRU 73356326 IC50 = 546000 nM T94033 COM4Q5 73356327 IC50 = 21000 nM T94033 CS7U3O 73356328 IC50 = 38000 nM T94033 CS06FN 73356329 IC50 = 109000 nM T94033 CW6ZD2 73356330 IC50 = 748000 nM T94033 C9ZYO5 73356332 IC50 = 1749000 nM T94033 CPEV49 73356333 IC50 = 25000 nM T94033 CFB57M 73356334 IC50 = 428000 nM T94033 C5V7DI 73356335 IC50 = 2500 nM T94033 C7A4BZ 73356336 IC50 = 406000 nM T94033 C5JBZ2 73356337 IC50 = 14000 nM T94033 C3I2HJ 73356338 IC50 = 51000 nM T94033 C8N4RM 73356390 Ki = 47 nM T94033 CYD8H6 73357220 Ki = 3.1 nM T94033 C94UWD 73357221 Ki = 0.29 nM T94033 CW6V3J 73357222 Ki = 0.25 nM T94033 C6BGR9 73604008 IC50 = 15500 nM T94033 CMS05I 75072534 Ki = 57 nM T94033 C5MVT3 76310068 Ki = 4400 nM T94033 CFH7S6 76310670 Ki = 6000 nM T94033 CD4AZ2 76311332 Ki > 100000 nM T94033 CS7WY0 76313442 Ki = 0.26 nM T94033 CUZM48 76314299 Ki = 3000 nM T94033 C6FQ0C 76314925 Ki = 353 nM T94033 CC2Q1D 76316954 Ki = 0.72 nM T94033 C54OUH 76316955 Ki = 80 nM T94033 CM3XH5 76316956 Ki = 0.13 nM T94033 C7QGZ9 76316957 Ki = 2.14 nM T94033 C9J0BH 76317785 Ki = 5600 nM T94033 CS92KW 76317870 IC50 > 44000 nM T94033 C9C4BV 76317871 Ki = 2000 nM T94033 CWH27L 76317872 Ki = 1000 nM T94033 CWZA05 76320988 Ki = 2900 nM T94033 C3BG6X 76321582 Ki = 6000 nM T94033 CP1MR4 76322205 Ki > 100000 nM T94033 CQN23P 76324323 Ki = 3.2 nM T94033 CSY7X9 76325187 Ki = 15000 nM T94033 COBF15 76325188 Ki = 3000 nM T94033 CO28RN 76325189 Ki = 2000 nM T94033 CQ98SD 76325190 Ki = 4000 nM T94033 CDB4R0 76325821 Ki > 100000 nM T94033 CP6HX3 76327889 Ki = 0.33 nM T94033 C2MEC1 76327890 Ki = 5 nM T94033 CJ10YI 76328088 IC50 = 390 nM T94033 C9O1BS 76328752 IC50 > 44000 nM T94033 CO3H5T 76328753 Ki = 14000 nM T94033 C1I2WQ 76328754 Ki = 3000 nM T94033 C59GFM 76328756 Ki = 1000 nM T94033 CZDM90 76331536 IC50 = 0.1 nM T94033 CYD98M 76331537 Ki = 2600 nM T94033 C6CW8M 76332426 Ki = 12000 nM T94033 C0BXZ8 76332427 Ki = 2000 nM T94033 CL6X7D 76335180 IC50 = 7 ug.mL-1 T94033 CO54FL 76336676 Ki = 69600 nM T94033 C10OJP 76336677 Ki = 17600 nM T94033 CAT95V 76685067 IC50 > 100000 nM T94033 CB6X5I 85735131 IC50 = 17600 nM T94033 CMD5V7 86583041 Ki > 12610 nM T94033 CV7IW5 87167024 Ki = 3985 nM T94033 CWP85J 87360663 IC50 = 62000 nM T94033 CO6U9I 88582319 Ki > 13300 nM T94033 CN4VU3 90643739 IC50 = 17000 nM T94033 C7DTZ4 90643740 IC50 = 13000 nM T94033 CYR29D 90643741 IC50 = 6500 nM T94033 CTJ7L8 90643744 IC50 = 8000 nM T94033 CTEH67 90643746 IC50 = 80000 nM T94033 CAY13O 90643748 IC50 = 20000 nM T94033 C6QO0I 90643751 IC50 = 30000 nM T94033 CT67GV 90643753 IC50 = 72000 nM T94033 CKC6Q3 90643754 IC50 = 20000 nM T94033 CA5S8R 90643757 IC50 = 15000 nM T94033 CKY0D3 90643758 IC50 = 4000 nM T94033 CT30UL 90643762 IC50 = 730 nM T94033 CJ6CN0 90644019 Ki = 2105 nM T94033 CB8KY3 90644020 Ki = 2852 nM T94033 C0G6SP 90644022 Ki = 501 nM T94033 CG83WX 90655748 Ki = 100000 nM T94033 CB68IT 90662976 IC50 = 350 nM T94033 C1RBK5 90663039 IC50 = 4000 nM T94033 CEL47S 90663088 IC50 = 36 nM T94033 CGEI71 90663100 IC50 = 50 nM T94033 C6LT7M 90663101 Ki = 110 nM T94033 C4J9FS 90663105 IC50 = 10000 nM T94033 CJP7F3 90663106 IC50 = 450 nM T94033 C4Q1FK 90663108 IC50 = 310 nM T94033 CF8SP9 90663109 IC50 = 160 nM T94033 C7TOZ2 90663110 IC50 = 39 nM T94033 CCSM17 90663112 IC50 = 10 nM T94033 CKH7W3 90663113 IC50 > 10000 nM T94033 CQ23MN 90663115 Ki = 70 nM T94033 CTK98I 90663126 IC50 = 260 nM T94033 CV62AS 90663132 IC50 = 38 nM T94033 CHUS10 90663138 IC50 = 12 nM T94033 CTC03D 90663139 IC50 = 13000 nM T94033 CV94QW 90663140 IC50 = 100 nM T94033 CP6A1S 90663152 IC50 = 600 nM T94033 CJS38O 90663164 IC50 = 11300 nM T94033 C6SK4I 90664135 IC50 > 1000 ug.mL-1 T94033 CE60BJ 90664137 IC50 > 1000 ug.mL-1 T94033 CYB39G 90664139 IC50 > 1000 ug.mL-1 T94033 C6KU0A 90664141 IC50 > 1000 ug.mL-1 T94033 C0D6LN 90664379 IC50 = 6.2 nM T94033 C7BX6R 90664760 Ki = 3 nM T94033 C0T4MS 90665251 IC50 > 1000 ug.mL-1 T94033 CD53HR 90665253 IC50 > 1000 ug.mL-1 T94033 CG32MX 90680086 IC50 = 1000 nM T94033 CVT5U6 90680087 IC50 = 10000 nM T94033 COH41Y 91666660 Ki > 13000 nM T94033 CA90QH 91827690 Ki = 11600 nM T94033 C5AC4V 101256535 Ki = 5 nM T94033 C65TLW 101862198 Ki > 1000000 nM T94033 C3PS6Y 118098650 Ki = 3800 nM T94033 C46MSP 118542774 Ki = 42300 nM T94033 C20WBY 118542785 Ki = 35900 nM T94033 CI65YK 118542879 Ki = 8100 nM T94033 CEH93P 118542958 Ki = 7400 nM T94033 CITU59 118548755 Ki > 100000 nM T94033 CMF5R6 118548758 Ki = 21900 nM T94033 C1IH2W 118548759 Ki > 100000 nM T94033 C6LZQ3 118548760 Ki > 100000 nM T94033 C62ZNW 118548761 Ki = 17000 nM T94033 C3WQ9D 118548776 Ki > 100000 nM T94033 CU01RP 118548813 Ki = 13400 nM T94033 CKS29X 118713018 IC50 > 100000 nM T94033 CRF62H 118713026 IC50 > 100000 nM T94033 CAS3L5 118713029 IC50 > 100000 nM T94033 C0GRU4 118718129 Ki = 0.007 nM T94033 CRV5Y1 118721008 Ki > 12610 nM T94033 C4U2AW 118723894 IC50 = 146000 nM T94033 CZ50SN 118723898 IC50 = 327000 nM T94033 CV5JG3 118723904 IC50 = 327000 nM T94033 CP98JL 118723906 IC50 = 425000 nM T94033 C0UO7Q 118723908 IC50 = 304000 nM T94033 CGL2B0 118725262 Ki = 794328.23 nM T94033 C3IA9S 118726913 IC50 > 20000 nM T94033 CABH86 118726934 IC50 > 20000 nM T94033 CO5X2B 118731971 IC50 = 48000 nM T94033 CVG2B0 118733057 IC50 = 5.86 nM T94033 C72UJV 118733058 IC50 = 6.166 nM T94033 CZLM10 118733059 IC50 = 4.93 nM T94033 CU9T2Y 118733060 IC50 = 4.786 nM T94033 CRGH87 118733061 IC50 = 4.571 nM T94033 C05QJD 118733062 IC50 = 16.22 nM T94033 CAL28Y 118733063 IC50 = 5.37 nM T94033 CX90OA 118733064 IC50 = 3.467 nM T94033 CR97IP 118733065 IC50 = 23.96 nM T94033 C8VU7G 118733066 IC50 = 5.623 nM T94033 C9OZ2B 118733067 IC50 = 7.244 nM T94033 C4T2RZ 118733068 IC50 = 21.38 nM T94033 C98DSY 118733109 IC50 = 3.71 nM T94033 CM4B3R 118733110 IC50 = 8.318 nM T94033 C1UK8R 118733111 IC50 = 4.92 nM T94033 CJ0B6R 118733112 IC50 = 23.44 nM T94033 CB3FZ7 118733113 IC50 = 4.898 nM T94033 CW5E8Q 118733114 IC50 = 13.49 nM T94033 CL0W6D 118733115 IC50 = 3.388 nM T94033 CV9NQ0 118733116 IC50 = 19.16 nM T94033 CJKV26 118736059 Ki = 1540000 nM T94033 C9TGN3 118736060 Ki = 1240000 nM T94033 C6EKO3 118736061 Ki = 580000 nM T94033 C5HYS2 118736062 Ki = 400000 nM T94033 C4M6UC 118736063 Ki = 370000 nM T94033 CI0H7T 118736064 Ki = 550000 nM T94033 CT8OW4 118736065 Ki = 512000 nM T94033 C7AT4H 118736067 Ki = 430000 nM T94033 C1G6JC 118736069 Ki = 370000 nM T94033 C86ECH 118736071 Ki = 136000 nM T94033 CCB41T 118736073 Ki = 76000 nM T94033 CT35WZ 118736075 Ki = 45000 nM T94033 CP5ZG1 118736077 Ki = 14000 nM T94033 CKEL03 118736078 Ki = 5000 nM T94033 CYH8F0 118736079 Ki = 3500 nM T94033 CQFJ53 118736080 Ki = 1000 nM T94033 C7MI6K 118736081 Ki = 1490 nM T94033 CNR78W 118736082 Ki = 220 nM T94033 CZ0R3W 118736083 Ki = 63000 nM T94033 CS45EX 118736084 Ki = 63000 nM T94033 CNYA31 118736085 Ki = 54000 nM T94033 C3U4YL 118736086 Ki = 54000 nM T94033 C7HJL0 118736088 Ki = 48000 nM T94033 C5JV7M 118736090 Ki = 22000 nM T94033 C2ZVQ6 118736092 Ki = 20000 nM T94033 C2M5CZ 118736094 Ki = 12000 nM T94033 C9JQP1 118736095 Ki = 600 nM T94033 CNZ68C 118736274 Ki = 140 nM T94033 C3D8RO 118736275 Ki = 40 nM T94033 CX38ZV 118736276 Ki = 10 nM T94033 C41AVK 118736277 Ki = 10 nM T94033 CC82LX 118736278 Ki = 27000 nM T94033 C3G9HC 118736280 Ki = 18000 nM T94033 C2H4PO 118736282 Ki = 20000 nM T94033 CB4U7V 118736284 Ki = 3600 nM T94033 C7Y1UR 118736286 Ki = 2600 nM T94033 CLC1P8 118736288 Ki = 1310 nM T94033 C9BKJ1 118753908 IC50 = 1.7 nM T94033 CHQ5P7 118987013 Ki > 12610 nM T94033 C5BUY6 119026228 IC50 = 800 nM T94033 C3NK4O 121232387 Ki = 2100 nM T94033 C3WC9Y 121488127 IC50 = 54000 nM T94033 C3YVQ8 122164611 Ki > 13300 nM T94033 CY1S5D 122164612 Ki > 13300 nM T94033 CKJN32 122164799 IC50 > 30000 nM T94033 C0IAV8 122182389 Ki = 499 nM T94033 CXT84D 122182390 Ki = 317 nM T94033 C3J7MH 122185884 IC50 = 5300 nM T94033 C8BK4F 122187244 Ki = 60 nM T94033 CP42JE 122192779 Ki > 50000 nM T94033 C43TNZ 122192780 Ki > 50000 nM T94033 C71IOQ 122192783 Ki = 381 nM T94033 CNJH01 122192784 Ki = 214 nM T94033 C9SDX8 122193065 IC50 = 9.2 nM T94033 C3Z2AP 122193309 IC50 = 4590 nM T94033 C16JAE 122194005 IC50 = 7.48 nM T94033 CG4LR5 122194707 Ki = 1900 nM T94033 C6NGM7 122194711 Ki = 3600 nM T94033 CR4CY8 122194712 Ki = 8600 nM T94033 C60ZMR 122194797 Ki = 270 nM T94033 CK94AY 122194799 Ki = 360 nM T94033 CD46TP 122194800 Ki = 57 nM T94033 C0KXN1 122194801 Ki = 590 nM T94033 C7AIC2 122194802 Ki = 65 nM T94033 C6J9KU 122194803 Ki = 8 nM T94033 CWJY13 122194804 Ki = 15 nM T94033 CR7MG0 122224465 IC50 > 500000 nM T94033 CAI69W 123238067 Ki = 29700 nM T94033 C76BAD 123424620 Ki = 2130 nM T94033 CK0W2P 127027635 Ki > 13000 nM T94033 CJ6DA9 127028140 IC50 > 10000 nM T94033 CD9KI3 127028141 IC50 > 10000 nM T94033 CPC0M8 127031390 Ki > 12610 nM T94033 CA30BN 127033248 Ki > 100000 nM T94033 CO7PY0 127033521 Ki > 100000 nM T94033 CE0QZ4 127033522 Ki = 82200 nM T94033 C7ZIR9 127034099 Ki > 100000 nM T94033 C1BWV2 127035672 Ki > 1000000 nM T94033 CVRY56 127036086 Ki > 1000000 nM T94033 C9B6LT 127037264 Ki > 1000000 nM T94033 C60HLK 127037469 Ki > 1000000 nM T94033 CQ98FX 127037729 IC50 = 199.53 nM T94033 CRIA10 127037730 IC50 = 26.3 nM T94033 C3BO8L 127038044 IC50 = 8.913 nM T94033 C5QYJ0 127038045 IC50 = 11.48 nM T94033 C5YA8I 127038046 IC50 = 10.96 nM T94033 C1RP2Z 127038047 IC50 = 39.81 nM T94033 CCE69I 127038048 IC50 = 36.31 nM T94033 C8OD5Q 127038110 IC50 = 117.49 nM T94033 CZ7MR3 127038111 IC50 = 2.042 nM T94033 CXTR41 127038454 IC50 = 28.18 nM T94033 CFWX25 127038455 IC50 = 18.62 nM T94033 CL3QG1 127039490 IC50 = 6.166 nM T94033 C8XV2L 127039491 IC50 = 9.55 nM T94033 CM1ZH8 127040121 IC50 = 117.49 nM T94033 C41POR 127040122 IC50 = 173.78 nM T94033 C0F3VT 127040123 IC50 = 17.38 nM T94033 CID14K 127040481 IC50 = 27.54 nM T94033 C4IYX8 127040482 IC50 = 26.92 nM T94033 C85ROH 127041472 IC50 > 100000 nM T94033 CQ7EL0 127042034 IC50 = 8.318 nM T94033 C53SCQ 127042068 IC50 = 23.99 nM T94033 CRL65F 127042754 IC50 = 3.69 nM T94033 C9M3NI 127042755 IC50 = 3.548 nM T94033 CMET26 127042756 IC50 = 7.413 nM T94033 C2Y0QA 127042759 IC50 = 4.266 nM T94033 CH01ZB 127042760 IC50 = 10.47 nM T94033 C8KX7Q 127042761 IC50 = 7.943 nM T94033 C9BEV2 127042983 IC50 = 12.3 nM T94033 CYH28P 127042984 IC50 = 3.95 nM T94033 C7PG6S 127042985 IC50 = 4.96 nM T94033 C90LJI 127045142 Ki = 15800 nM T94033 C4T9KU 127045502 Ki = 7400 nM T94033 C4RFP7 127045503 Ki > 11500 nM T94033 C2IOG9 127045504 Ki > 11500 nM T94033 CHK80O 127045505 Ki > 11500 nM T94033 CL6W5N 127045506 Ki > 11500 nM T94033 C80UJD 127045704 IC50 = 4.898 nM T94033 CW4JN5 127045705 IC50 = 7.18 nM T94033 CA3SB2 127045706 IC50 = 5.66 nM T94033 CJ1S0F 127045707 IC50 = 1.81 nM T94033 CSM92B 127045729 IC50 = 4.169 nM T94033 C78QIO 127045731 IC50 = 3.21 nM T94033 CRZ3E2 127045911 IC50 = 5.44 nM T94033 C3ZT9X 127045918 IC50 = 10.05 nM T94033 C1IPX7 127045944 IC50 = 9.12 nM T94033 CVRG73 127046181 IC50 = 2.16 nM T94033 COPY57 127053575 Ki = 0.15 nM T94033 C4CB3A 129012067 Ki = 9.2 nM T94033 CM2A6S 129012068 Ki = 0.07 nM T94033 C90XNU 129824058 IC50 = 3.35 nM T94033 CW7A4U 129824062 IC50 = 1.54 nM T94033 CE26HW 131955087 IC50 = 94000 nM T94033 CT2RV6 134130781 IC50 > 1000000 nM T94033 CWV3G6 134131077 IC50 > 200000 nM T94033 CS8FV1 134131084 IC50 > 200000 nM T94033 C92RTL 134131303 IC50 > 200000 nM T94033 CL37SG 134131589 IC50 > 200000 nM T94033 CPQ04R 134132204 Ki > 10000 nM T94033 CA8E6Z 134132206 IC50 = 82.8 nM T94033 CC7UO1 134133660 Ki > 13300 nM T94033 CRA07M 134135715 IC50 = 3.11 nM T94033 C9VI1D 134135793 IC50 = 2.13 nM T94033 C3ZRP2 134137891 IC50 = 1002 nM T94033 C17RCM 134138069 IC50 = 4.98 nM T94033 C9Z4TV 134139904 IC50 = 437 nM T94033 C6DPW7 134141496 Ki > 10000 nM T94033 C4X7UQ 134142073 IC50 = 6.27 nM T94033 C9RW1V 134142735 IC50 = 456 nM T94033 CGL60E 134144735 IC50 = 3.1 nM T94033 C3IN2W 134144920 IC50 = 1.62 nM T94033 CIRU10 134145163 Ki = 9000 nM T94033 CHA7X9 134146314 Ki > 10000 nM T94033 C5Y9DL 134146919 IC50 = 446 nM T94033 CS05TI 134148116 IC50 = 6.59 nM T94033 C9UZI0 134148669 Ki = 18000 nM T94033 CTG65U 134148771 Ki > 10000 nM T94033 CRWO87 134148886 IC50 = 16.45 nM T94033 CR6V9U 134150310 Ki > 13300 nM T94033 CKBZ10 134151065 IC50 = 1440 nM T94033 CMGR41 134151623 IC50 = 1925 nM T94033 C3QEO5 134151811 Ki > 10000 nM T94033 C9FMR2 134151871 IC50 = 1028 nM T94033 CUWZ32 134153767 IC50 = 4.69 nM T94033 C43XLC 134154061 IC50 = 147 nM T94033 CKGD09 134154240 IC50 = 0.92 nM T94033 CV0RS5 134156046 IC50 = 511 nM T94033 CG9UL4 134156593 Ki > 13300 nM T94033 C2YVB4 134157252 IC50 = 4.23 nM T94033 CD06PE 134313025 IC50 > 20000 nM T94033 C6HTD5 135393470 IC50 > 10000 nM T94033 C7NA6E 135393474 IC50 > 20000 nM T94033 CBW03G 135404142 Ki > 5000 nM T94033 C8GE5V 135404808 Ki = 680 nM T94033 CD53CZ 135404951 Ki > 4000 nM T94033 C9YUQ1 135405121 Ki = 2280 nM T94033 C9SY8U 135406499 Ki = 1400 nM T94033 CQEZ96 135406539 Ki > 4000 nM T94033 C94GZP 135406646 Ki = 190 nM T94033 CP7Z3S 135407592 Ki = 650 nM T94033 C5XA6H 135407717 Ki = 38000 nM T94033 C0OX6T 135407736 Ki = 34000 nM T94033 CA8X0V 135409826 Ki = 190 nM T94033 CD48MU 135415156 Ki = 490 nM T94033 CNIE32 135426905 Ki = 4500 nM T94033 CK1AD7 135426949 Ki = 280 nM T94033 C61XOA 135427245 Ki = 80000 nM T94033 CL25SO 135427324 Ki = 880 nM T94033 C2I6WX 135430716 Ki > 150000 nM T94033 CHMD42 135431470 Ki = 44000 nM T94033 C8WS4O 135443730 Ki = 65000 nM T94033 CTP5V8 135444609 Ki = 15000 nM T94033 C3SMN4 135444666 IC50 > 10000 nM T94033 C4M5BF 135450980 Ki > 75000 nM T94033 CKA3D2 135451808 Ki = 630 nM T94033 CDT1C6 135452907 Ki = 2.5 nM T94033 C3YT2M 135452929 Ki = 3 nM T94033 CPN5I3 135452944 Ki = 0.02 nM T94033 C9KLD3 135455964 Ki = 2000 nM T94033 CSK06Y 135456121 Ki = 57800 nM T94033 CJWC64 135462427 Ki = 206 nM T94033 CP30YA 135469657 Ki = 26 nM T94033 C5O6JX 135469686 Ki = 0.05 nM T94033 C9XMA6 135469687 Ki = 0.05 nM T94033 CXS6B9 135471524 Ki = 17000 nM T94033 C5PO0Q 135471605 Ki = 3400 nM T94033 CU8IC7 135474643 Ki = 5100 nM T94033 C2PFI8 135475618 Ki = 1100 nM T94033 CI8Z4U 135479981 Ki = 1200 nM T94033 CG2N5B 135484079 Ki = 0.2 nM T94033 C50EKI 135484100 Ki > 5000 nM T94033 CBE9G0 135490854 Ki = 80000 nM T94033 CZGI04 135490911 Ki = 120 nM T94033 CPE5Y8 135490928 IC50 = 575.44 nM T94033 C9T1IA 135492878 Ki > 5000 nM T94033 CRNB95 135492887 Ki > 5000 nM T94033 CPW07U 135493126 Ki = 0.17 nM T94033 C9TA2B 135501173 Ki = 250 nM T94033 CO5UV8 135501194 Ki = 140 nM T94033 CMQ6O0 135501618 Ki = 48000 nM T94033 C47UGJ 135503965 Ki = 2219 nM T94033 C0NS9U 135506896 Ki = 15 nM T94033 CH5AN0 135509745 IC50 = 288.4 nM T94033 CVA61N 135512760 Ki = 37000 nM T94033 CLO72H 135514651 Ki = 710 nM T94033 CP51ZM 135515290 Ki = 125 nM T94033 CW7TI2 135515464 Ki > 10000 nM T94033 C3MLP1 135517489 Ki > 5000 nM T94033 CLFR21 135528485 Ki = 0.51 nM T94033 CHEQ21 135528490 Ki = 2.1 nM T94033 CL8PD0 135528527 Ki = 0.63 nM T94033 CSW47P 135528873 Ki = 90000 nM T94033 CET9Q2 135530746 Ki > 21000 nM T94033 C4OW8A 135531345 Ki = 192 nM T94033 CK97FT 135533257 Ki = 12000 nM T94033 CAD75F 135535997 Ki = 70000 nM T94033 C3E4CU 135537603 Ki = 1100 nM T94033 C6UH2Y 135542698 IC50 = 134.9 nM T94033 C67TIA 135544099 IC50 > 10000 nM T94033 CDT59O 135544137 Ki = 2800 nM T94033 CCH49A 135544551 Ki = 7000 nM T94033 CKLD47 135544579 Ki = 90000 nM T94033 CSO35D 135546147 Ki > 5000 nM T94033 C5RG6Z 135546170 Ki = 810 nM T94033 CD9AO5 135548205 Ki = 180 nM T94033 C7Q9YK 135559071 Ki > 150000 nM T94033 CAU8S4 135559072 Ki > 150000 nM T94033 C69ZVL 135559080 Ki = 15 nM T94033 C9D1MQ 135581665 Ki = 890 nM T94033 CB6L5Y 135581668 Ki = 5140 nM T94033 C5ZFS3 135581673 Ki > 5000 nM T94033 CYG47F 135581674 Ki > 5500 nM T94033 C94JBX 135581677 Ki = 480 nM T94033 C05ONT 135581679 Ki = 250 nM T94033 CUL71O 135581680 Ki = 1100 nM T94033 C5YW3X 135581684 Ki = 1820 nM T94033 C09QFL 135667566 Ki = 1300 nM T94033 CGE51P 135672692 IC50 >= 30000 nM T94033 C8KNC4 135681488 Ki = 0.06 nM T94033 C58PSA 135740053 Ki > 6000 nM T94033 C4VL1K 135740054 Ki > 6000 nM T94033 CZL58Y 135740055 Ki > 6000 nM T94033 CR05YT 135740056 Ki > 6000 nM T94033 C2O7PT 135740057 Ki > 6000 nM T94033 C6MZP7 135763271 Ki > 4000 nM T94033 C68GTN 135763273 Ki = 3200 nM T94033 C91UXW 135802775 Ki > 4000 nM T94033 C0AX3J 135802853 Ki > 5000 nM T94033 CRB42G 135802854 Ki = 1000 nM T94033 CQD2Z1 135855944 Ki = 4.2 nM T94033 CMJ0B6 135962022 Ki > 4000 nM T94033 C4MU7I 135964427 Ki = 0.42 nM T94033 C39BCV 135964431 Ki < 0.01 nM T94033 CIL54R 135964432 Ki = 0.08 nM T94033 C7YVL9 135981708 IC50 > 50000 nM T94033 CC54EI 135986123 IC50 = 27.96 nM T94033 C9G7TE 135995982 Ki = 350 nM T94033 C84ZQA 135998835 Ki = 0.24 nM T94033 CE1F4K 136029159 Ki = 560 nM T94033 CK36ZW 136029160 Ki = 0.13 nM T94033 CV16LS 136032597 Ki = 0.09 nM T94033 C6S5OL 136034781 Ki = 50000 nM T94033 CPSO31 136045813 Ki > 10000 nM T94033 CYQ70K 136053621 IC50 > 11000 nM T94033 C46VRO 136058172 Ki = 2900 nM T94033 C6Q4FB 136058174 Ki > 4000 nM T94033 C34UZI 136058175 Ki > 4000 nM T94033 CUX79V 136058176 Ki > 4000 nM T94033 CBY56D 136058177 Ki > 4000 nM T94033 C4YO6Q 136058178 Ki ~ 4000 nM T94033 CB39EK 136058180 Ki > 4000 nM T94033 C8PLB3 136058181 Ki > 4000 nM T94033 CSU6X4 136058182 Ki > 4000 nM T94033 C0Y3CA 136058183 Ki > 4000 nM T94033 C8IH1Z 136058184 Ki > 4000 nM T94033 C4LG7S 136058185 Ki > 4000 nM T94033 CCX30L 136058186 Ki > 4000 nM T94033 C6KG8F 136058187 Ki > 4000 nM T94033 CHS25L 136058188 Ki > 4000 nM T94033 C8G4TI 136066129 Ki > 6000 nM T94033 CY6XD7 136066130 Ki > 6000 nM T94033 CN70IU 136092208 Ki > 75000 nM T94033 C5N3KP 136092209 Ki = 10000 nM T94033 C1BUH6 136092210 Ki = 50000 nM T94033 CFQ2C8 136092211 Ki = 22000 nM T94033 CX5R9J 136092212 Ki = 14000 nM T94033 C35PXN 136092213 Ki = 32000 nM T94033 CEXJ30 136092214 Ki > 75000 nM T94033 CS6QH0 136092215 Ki = 165000 nM T94033 CMR7L4 136092216 Ki = 70000 nM T94033 CN0WR7 136092217 Ki = 20000 nM T94033 COCN35 136092218 Ki = 20000 nM T94033 CA79JC 136092219 Ki = 31000 nM T94033 CA2TD8 136094852 IC50 = 57.4 nM T94033 CQW40T 136104458 IC50 > 100000 nM T94033 CI7XJ3 136104459 IC50 > 100000 nM T94033 CSP4A7 136114639 Ki = 210 nM T94033 CPK6X2 136198635 Ki = 920 nM T94033 CRJ5S4 136198636 Ki = 2600 nM T94033 C7WE2G 136198637 Ki = 4000 nM T94033 C12UWY 136198638 Ki = 2600 nM T94033 CT1QN2 136224837 Ki > 100000 nM T94033 CN8BW0 136224847 Ki > 100000 nM T94033 C7KE9J 136224848 Ki > 100000 nM T94033 C7R1TS 136224849 Ki > 100000 nM T94033 CG24CQ 136224854 Ki > 100000 nM T94033 C9QCG6 136236347 Ki = 0.09 nM T94033 C3FRZ4 137629177 Ki = 340 nM T94033 C2JT1W 137632528 IC50 = 267000 nM T94033 CZ7PN0 137632696 Ki = 4200 nM T94033 CU4ZC5 137633305 Ki = 11900 nM T94033 CSR3A2 137635035 Ki = 68000 nM T94033 CYUW38 137635103 Ki = 250000 nM T94033 CDQ62V 137637214 Ki > 50000 nM T94033 C6JX1F 137637665 IC50 = 14.6 nM T94033 C2K8JV 137639385 Ki > 50000 nM T94033 C7CG5Z 137639572 Ki = 17900 nM T94033 C4UHF8 137641581 IC50 = 12.77 nM T94033 CLA6B3 137642880 Ki = 4000 nM T94033 C6UO7S 137643149 IC50 = 0.84 nM T94033 C19GEB 137643298 Ki = 44000 nM T94033 C7YI0J 137643322 IC50 = 67000 nM T94033 CH26WY 137644461 Ki = 163000 nM T94033 CNO2T8 137647340 IC50 = 156000 nM T94033 CJK39I 137648564 Ki = 59000 nM T94033 CQ6J1M 137650284 Ki = 14500 nM T94033 CCL27W 137650547 IC50 = 3.7 nM T94033 C6WVH7 137651104 IC50 = 2.26 nM T94033 CVC4G9 137652563 IC50 = 81000 nM T94033 CGC01N 137653173 Ki = 68000 nM T94033 CA6X7H 137654486 IC50 = 1.18 nM T94033 CNX46H 137654508 Ki > 50000 nM T94033 CZ1H4R 137655362 Ki > 10000 nM T94033 CN83KL 137657877 Ki = 36000 nM T94033 C5B6AF 137658068 Ki = 7100 nM T94033 CAJP67 137658480 IC50 = 3.2 nM T94033 CWO8D4 137659456 Ki = 13500 nM T94033 CIQV31 137661258 IC50 = 1.42 nM T94033 CK4C7O 137797022 Ki = 3.51 nM T94033 CUZ35A 138115400 IC50 = 63095.73 nM T94033 CO51HN 139030452 IC50 > 20000 nM T94033 C6LG0F 139589789 IC50 = 250000 nM T94033 CX07YE 139592452 Ki > 13300 nM T94033 C0T6OH 140430655 Ki = 483.63 nM T94033 C0A3MI 145959466 IC50 > 50000 nM T94033 CC8O5G 145963849 IC50 = 1300 nM T94033 C9WAO7 145964010 IC50 = 2300 nM T94033 CE5M2N 145964487 IC50 > 300000 nM T94033 CNHT51 145964676 IC50 = 134000 nM T94033 CZH21Q 145965556 IC50 > 500000 nM T94033 C78LKX 145966681 IC50 > 300000 nM T94033 CC3XB0 145967211 IC50 = 2600 nM T94033 C8FGZ3 145968728 IC50 = 3200 nM T94033 C1ZU9C 145968968 IC50 = 1300 nM T94033 C1WAP5 145969641 IC50 > 500000 nM T94033 C62OHZ 145970288 IC50 = 134000 nM T94033 CE6C0A 145970642 Ki = 10600 nM T94033 CRNW09 145971341 IC50 = 4000 nM T94033 CSA3U0 145971563 IC50 = 8700 nM T94033 C9CH7V 145972272 IC50 = 3800 nM T94033 CE1M4I 145972287 IC50 = 2600 nM T94033 CN08VA 145972739 IC50 = 168000 nM T94033 CNQ47U 145973701 IC50 = 2000 nM T94033 CS1N3E 145974035 IC50 = 229000 nM T94033 CJN59A 145974171 IC50 > 500000 nM T94033 C6J0YW 145974544 IC50 = 250000 nM T94033 CH5G9E 145975062 IC50 = 3300 nM T94033 CUG23Y 145975277 IC50 > 500000 nM T94033 C5GL0V 145975446 IC50 > 500000 nM T94033 C8N4YW 145975510 IC50 = 4900 nM T94033 CN8K3X 145975689 IC50 = 2600 nM T94033 CJU6V7 145976287 IC50 = 2600 nM T94033 COM3R1 145976303 IC50 > 500000 nM T94033 CGFZ02 145977247 IC50 = 100000 nM T94033 C1JS9L 145977781 IC50 > 500000 nM T94033 CGCA85 145978637 IC50 > 500000 nM T94033 C2JF8N 145978807 IC50 = 14000 nM T94033 C4HLX8 146029523 IC50 > 20000 nM T94033 CSBC71 146680900 IC50 = 27000 nM T94033 CJP64T 155510867 IC50 > 20000 nM T94033 CZR36C 155511554 IC50 = 10000 nM T94033 C2VX3G 155512946 Ki > 11500 nM T94033 CYT20V 155514020 Ki > 50000 nM T94033 CAT98N 155514640 Ki > 10000 nM T94033 C8WR1O 155515070 Ki = 310 nM T94033 C37MUL 155515203 IC50 = 4.2 nM T94033 CPUG37 155516479 Ki = 4.6 nM T94033 CF96DM 155518671 Ki > 10000 nM T94033 C6NX4K 155519661 IC50 = 3981.07 nM T94033 C4MS1B 155519676 IC50 = 15848.93 nM T94033 C7DUX3 155520916 Ki > 10000 nM T94033 CE01NY 155523107 IC50 > 20000 nM T94033 CW9K3R 155523263 IC50 > 20000 nM T94033 CGMP07 155523803 IC50 > 20000 nM T94033 CBU5W0 155524880 IC50 > 10000 nM T94033 CN3BH5 155527998 IC50 = 3162.28 nM T94033 CR84UG 155528520 Ki = 360 nM T94033 CHYW65 155528639 IC50 = 1995.26 nM T94033 CG68UH 155529134 IC50 > 20000 nM T94033 CD7O2G 155530095 IC50 = 10000 nM T94033 CA82SM 155530516 Ki = 1618 nM T94033 C46AZL 155530642 Ki > 25000 nM T94033 C35QWO 155531023 IC50 = 19952.62 nM T94033 C2X5EJ 155531124 IC50 > 10000 nM T94033 CL1PN0 155531210 Ki = 1213 nM T94033 C3AL6D 155533619 IC50 = 32 nM T94033 CY3FE6 155533938 IC50 = 7.1 nM T94033 C7M2UT 155534310 IC50 > 20000 nM T94033 C12HON 155536142 IC50 = 19952.62 nM T94033 C1V9GL 155538855 Ki = 140 nM T94033 CC9EY4 155538891 Ki = 490 nM T94033 CL90DN 155540666 Ki > 10000 nM T94033 CY6DK3 155540964 IC50 = 398.11 nM T94033 CAT09J 155541500 Ki = 200 nM T94033 CR12YK 155542064 Ki = 200 nM T94033 C4P2GV 155543617 Ki > 25000 nM T94033 CT4S3M 155544624 IC50 > 20000 nM T94033 CY7DK3 155545696 Ki = 260 nM T94033 CM9TA0 155545734 Ki = 190 nM T94033 CU52QS 155545897 Ki > 10000 nM T94033 CQ51DI 155546002 IC50 = 7700 nM T94033 CH2S6R 155546346 Ki > 10000 nM T94033 C5MB9R 155547962 IC50 = 3162.28 nM T94033 C0D5YW 155548172 IC50 > 2000 nM T94033 CLFB25 155548371 IC50 = 6309.57 nM T94033 CWC8X9 155550748 IC50 > 100000 nM T94033 C4XP1J 155551078 Ki = 117000 nM T94033 CU9FL4 155551858 Ki > 50000 nM T94033 COM52R 155551892 IC50 = 1995.26 nM T94033 C7SE3N 155553319 Ki = 3400 nM T94033 CJ3FI5 155553630 IC50 = 31622.78 nM T94033 C2E5GR 155554478 IC50 > 10000 nM T94033 CYT86P 155554873 Ki = 28 nM T94033 CU8LR3 155555208 Ki > 25000 nM T94033 CE3G5W 155556110 IC50 > 10000 nM T94033 C0SND3 155557259 IC50 > 10000 nM T94033 CSW48V 155557718 IC50 = 1258.93 nM T94033 CR4FE5 155557809 Ki = 2700 nM T94033 CTS63Q 155558248 IC50 > 10000 nM T94033 CFX07G 155558369 IC50 > 10000 nM T94033 CWF3C9 155558681 Ki = 2500 nM T94033 C1HTZ4 155559077 IC50 = 530 nM T94033 C5ST1B 155559602 Ki = 379 nM T94033 CNZ1K5 155559920 Ki > 10000 nM T94033 C0FWQ1 155564112 Ki = 500 nM T94033 C2AM3T 155564229 Ki = 50 nM T94033 CM8XB1 155565537 IC50 = 2511.89 nM T94033 CTF0S7 155566456 Ki = 2948 nM T94033 C7WQJ3 155567187 Ki = 57 nM T94033 CP4F1U 155567613 Ki > 50000 nM T94033 C13NDJ 155567925 Ki = 12000 nM T94033 CEZ8B9 155568406 Ki > 50000 nM T94033 C95JMP 10135437 Ki = 1.9 nM T94033 CRM13Y 10225608 Ki = 1 nM T94033 C2GES3 2037 IC50 = 10 ug.mL-1 T94033 C2EIA8 44287957 Ki = 4.9 nM T94033 C9TO4H 44288242 Ki = 4.7 nM T94033 CEJ04P 44337861 IC50 = 310 nM T94033 C76YMC 44337909 IC50 = 16 nM T94033 C4VKN5 44337910 IC50 = 55 nM T94033 C2TFX8 44337951 IC50 = 43 nM T94033 CQ3G8A 44337952 IC50 = 19 nM T94033 CI5BX0 44337970 IC50 = 230000 nM T94033 CWNK26 44337971 IC50 = 19 nM T94033 CNC73Z 44338047 IC50 = 8.3 nM T94033 CVK8X3 44338049 IC50 = 0.008 nM T94033 CD81GH 46830813 IC50 > 2500 nM T94033 D00KJP 10322586 Ki = 1000 nM T94033 D00WFQ 674641 IC50 = 12100 nM T94033 D01ARY 44405865 Ki = 0.5 nM T94033 D01LCS 447480 Ki = 15000 nM T94033 D01NEZ 16079152 IC50 = 5.8 nM T94033 D01RTU 448763 Ki = 4.9 nM T94033 D02AVL 18376720 Ki = 990 nM T94033 D02KKL 1282 Ki = 1 nM T94033 D02NHS 154118 Ki = 0.8 nM T94033 D02PAU 16731825 Ki = 3700 nM T94033 D02XPB 23646462 Ki = 270 nM T94033 D02YIW 1794 IC50 > 10000 nM T94033 D03QAQ 9869498 Ki = 300 nM T94033 D03ZUM 6917805 IC50 = 45 nM T94033 D05ICF 3492365 IC50 = 2300 nM T94033 D05ZIP 674656 IC50 = 4700 nM T94033 D06GTS 76318115 IC50 >= 30000 nM T94033 D06HOI 44249821 Ki = 6600 nM T94033 D06KCW 6323178 IC50 = 130 nM T94033 D06LPR 674651 IC50 = 11900 nM T94033 D06MTX 1506 Ki = 55000 nM T94033 D07IBU 10696098 IC50 = 4 nM T94033 D07SFI 2332 Ki = 300 nM T94033 D07SGS 44292136 Ki = 7900 nM T94033 D07ZRG 46899577 Ki = 1.94 nM T94033 D08EUH 25113125 Ki = 4600 nM T94033 D08OCS 699665 IC50 = 4300 nM T94033 D08WQJ 700133 IC50 = 11000 nM T94033 D09OBJ 9872263 Ki = 0.18 nM T94033 D0A8WP 447732 Ki = 5600 nM T94033 D0C1TS 44272875 Ki = 0.14 nM T94033 D0CF3B 44584173 IC50 = 67.9 nM T94033 D0CT8A 23646461 Ki = 4500 nM T94033 D0CV4F 44405859 Ki = 36 nM T94033 D0D8AK 44584171 IC50 = 2.9 nM T94033 D0F2YC 10038543 IC50 = 72 nM T94033 D0F6EZ 44436702 Ki > 1000000 nM T94033 D0H5WV 5289082 IC50 = 28 nM T94033 D0I0NY 10322542 Ki = 0.09 nM T94033 D0IU5E 716930 IC50 = 390 nM T94033 D0J1CC 11948634 Ki > 15000 nM T94033 D0J1QT 44473100 Ki = 2300 nM T94033 D0J2SM 296008 IC50 = 510 nM T94033 D0JU9N 6914623 Ki = 35 nM T94033 D0K7YL 447476 Ki = 320 nM T94033 D0M1AC 44584172 IC50 = 7.4 nM T94033 D0M1LO 205051 Ki = 150 nM T94033 D0M4VZ 10456438 IC50 = 2500 nM T94033 D0MQ6K 10574241 Ki > 4000 nM T94033 D0O0GT 44272797 Ki = 0.56 nM T94033 D0O1DU 25011732 Ki = 90 nM T94033 D0ON2Z 204102 Ki = 540 nM T94033 D0R4AV 5288064 Ki = 0.24 nM T94033 D0R5KV 4322 Ki = 2000 nM T94033 D0R9CH 3400921 Ki = 90 nM T94033 D0RQ2T 44331282 Ki = 4.1 nM T94033 D0SP2I 6852210 Ki = 110 nM T94033 D0T5WR 44405684 Ki = 66 nM T94033 D0T9WZ 54613196 IC50 >= 30000 nM T94033 D0U4HG 23634523 IC50 = 12300 nM T94033 D0V3PG 128861 IC50 = 250 nM T94033 D0V6DX 10640 IC50 > 5000 nM T94033 D0V7AA 9064 IC50 = 125000 nM T94033 D0V7RD 10439038 IC50 = 46 nM T94033 D0V7TH 76328755 Ki = 500 nM T94033 D0W2SV 70689167 Ki = 637 nM T94033 D0X0IF 23655936 IC50 = 17800 nM T94033 D0X1OY 674628 IC50 = 2800 nM T94033 D0Y5IQ 44255320 IC50 = 10000 nM T94033 D0Y8QU 9869156 Ki = 1 nM T94033 D0Y9PH 45486355 Ki = 23000 nM T03644 C5EUF4 7108 Ki > 500 nM T03644 CY9M6K 61365 IC50 = 322000 nM T03644 CAG41Z 621196 Ki = 121.8 nM T03644 CO41FC 964143 Ki = 290.2 nM T03644 CO1ZV8 2306524 Ki = 206.7 nM T03644 CTNQ85 3838042 Ki = 116.5 nM T03644 CY28LS 5293755 Ki = 507.6 nM T03644 C5ZS3K 5713403 Ki = 621.8 nM T03644 CZ9Q1O 5928757 Ki = 347.2 nM T03644 CQ3S8L 6450842 Ki = 84.4 nM T03644 CFXW58 11631766 Ki = 959.3 nM T03644 CDQC89 21254490 Ki > 500 nM T03644 CDN1A2 44555764 Ki > 500 nM T03644 CU1D5F 58795397 Ki = 144.4 nM T03644 CQU9W0 66556402 Ki = 124.3 nM T03644 CU9ZN4 70684415 Ki > 500 nM T03644 C1SWK5 70686556 Ki = 106 nM T03644 C7BY9N 70686557 Ki > 500 nM T03644 CQ15TA 70686558 Ki > 500 nM T03644 CF0M8T 70686559 Ki > 500 nM T03644 C3UQ8O 70688673 Ki > 500 nM T03644 C59SNL 70688674 Ki = 57.9 nM T03644 CWK41G 70688675 Ki > 500 nM T03644 CU8C9X 70690739 Ki = 346 nM T03644 CMF80G 70690740 Ki = 32.1 nM T03644 CJC2D8 70692879 Ki = 75.3 nM T03644 CM3UQ6 70692880 Ki = 49 nM T03644 CD2MY5 70696968 Ki > 500 nM T03644 CTA8R4 90662826 Ki > 500 nM T03644 CB03DR 122182244 Ki = 407.1 nM T03644 CI6WT0 122182245 Ki = 114.5 nM T03644 C3X5KJ 122182246 Ki = 149.8 nM T03644 CT5G1Q 122182247 Ki = 342.6 nM T03644 CCT7H6 122182248 Ki = 350.2 nM T03644 CML3T5 122182249 Ki = 79.5 nM T03644 CMO1C3 122182250 Ki = 61.1 nM T03644 CIT52U 122182251 Ki = 40.7 nM T03644 C19GJH 122182252 Ki = 11.5 nM T03644 CUOB01 122182253 Ki = 54 nM T03644 CW2V5B 122182254 Ki = 226.9 nM T03644 C75OCP 122182255 Ki = 72.5 nM T03644 CVH2T0 122182256 Ki = 63.7 nM T03644 CKQF12 122182257 Ki = 40.9 nM T03644 C7AUF8 122182258 Ki = 54.6 nM T03644 C7BXY4 122182259 Ki = 4.2 nM T03644 CCEL74 122182260 Ki = 92 nM T03644 C32GEV 122182261 Ki = 45.3 nM T03644 CWIT38 122182262 Ki = 68.3 nM T03644 CMVS36 122182263 Ki = 29.8 nM T03644 CLW95X 122182264 Ki = 43.6 nM T03644 C4TNB1 122182265 Ki = 68.1 nM T03644 CQ4R0K 122182266 Ki = 44.8 nM T03644 C5C8FY 122182267 Ki = 482.9 nM T03644 C7NV9G 122182268 Ki = 14.6 nM T03644 CU3NJ6 122182269 Ki = 211.4 nM T03644 CS84HC 122182270 Ki = 25 nM T03644 C8EYO3 122182271 Ki = 192.7 nM T03644 CFV32E 122182272 Ki = 12.9 nM T03644 C1LHQ2 122182273 Ki = 81.9 nM T03644 C24PHB 122182274 Ki = 3.8 nM T03644 C1U3FZ 122182275 Ki = 64.7 nM T03644 CX5NB4 122182276 Ki = 3.5 nM T03644 CAU9H6 122182277 Ki = 53.3 nM T03644 C2RB1F 122182278 Ki = 2.1 nM T03644 CTMV35 122182279 Ki = 76.1 nM T03644 C6Y5OP 135262740 IC50 = 3200 nM T03644 CQD78E 135263240 IC50 = 4600 nM T03644 C9VGZ4 135263274 IC50 = 1900 nM T03644 C3FVU2 135263287 IC50 = 3700 nM T03644 C7SO3K 155510664 IC50 = 2190 nM T03644 CL4XJ9 155516842 IC50 = 3130 nM T03644 CX0TR5 155530957 IC50 = 4430 nM T03644 CV1U2Z 155553595 IC50 = 1850 nM T03644 C2PJ7U 155555711 IC50 = 1090 nM T03644 CM9ZE2 155557325 IC50 = 2050 nM T03644 D0H2MA 6324599 IC50 = 5400 nM T17036 D0BA6T 38853 IC50 = 3000 nM T17036 D0E7PQ 5311 IC50 = 540000 nM T17036 D0R6BI 3341 Ki = 1920 nM T17036 D0T7OW 681 IC50 = 3000 nM T17036 D0W0VD 3885 IC50 = 3000 nM T17036 D00SUC 74766595 IC50 = 160 nM T17036 D03TPE 97394 IC50 = 2000 nM T17036 D09NCT 53392492 IC50 = 5900 nM T17036 D0WC4Z 45376646 IC50 = 5000 nM T17036 CWJ0U1 5312 IC50 = 23900 nM T17036 CVZ1A0 38101 Ki = 1980 nM T17036 C06WZQ 222878 IC50 = 200 nM T17036 COS62U 245007 IC50 > 100000 nM T17036 C0MHV8 252439 IC50 = 400 nM T17036 CU08TX 279619 IC50 = 11000 nM T17036 C5K3ZJ 459531 IC50 = 1258.93 nM T17036 CBN91O 655278 IC50 = 1100 nM T17036 C2OS3W 2238068 IC50 > 100000 nM T17036 CEQ4V8 2723716 IC50 > 100000 nM T17036 CTC90M 6519698 IC50 = 316.23 nM T17036 CCYF63 9942424 IC50 = 398.11 nM T17036 C30EMN 24701909 IC50 = 4800 nM T17036 CF47JU 25138011 IC50 = 5000 nM T17036 C7X3WA 28330466 IC50 > 100000 nM T17036 CO18LM 45104128 IC50 = 200000 nM T17036 CP59WA 45376516 IC50 = 5400 nM T17036 C1WL2X 45376644 IC50 = 5000 nM T17036 C1KPR6 45377880 IC50 = 180 nM T17036 CTIN21 45378188 IC50 = 110 nM T17036 C0HCX8 50916282 IC50 = 2500 nM T17036 CJ6D9P 56663048 IC50 = 200000 nM T17036 CL3HT1 71449736 IC50 > 100000 nM T17036 CJH86V 71451542 IC50 > 100000 nM T17036 CH38AO 71453382 IC50 > 100000 nM T17036 C2U4AQ 71458738 IC50 = 4300 nM T17036 CYF8O7 71767874 IC50 = 39.81 nM T17036 C68RKH 76310231 IC50 = 3900 nM T17036 CO1EN3 76317452 IC50 = 420 nM T17036 CT5FZ8 76321184 IC50 = 5500 nM T17036 C6XRT0 76321186 IC50 = 16000 nM T17036 CKB5O9 76328366 IC50 = 5100 nM T17036 CUNK03 76335652 IC50 = 3500 nM T17036 C63ATV 81750201 IC50 = 39.81 nM T17036 CIG3E9 83672127 IC50 = 13000 nM T17036 C83TUW 89825693 IC50 = 50.12 nM T17036 C2NA5I 91801131 IC50 = 15848.93 nM T17036 C10RDJ 101882871 IC50 > 100000 nM T17036 C86LNW 101882872 IC50 > 100000 nM T17036 C4FPD3 112726150 IC50 > 100000 nM T17036 C8E2KI 122191450 IC50 = 6309.57 nM T17036 C75JVN 122191451 IC50 = 79432.82 nM T17036 C3YX7W 122191453 IC50 = 79432.82 nM T17036 C3IBR8 122191455 IC50 = 50118.72 nM T17036 C59KNQ 122191457 IC50 > 100000 nM T17036 CM5X8J 122191459 IC50 = 100000 nM T17036 C7ASR0 122191460 IC50 > 100000 nM T17036 CRI6J4 122191461 IC50 > 100000 nM T17036 CAS4H6 122191462 IC50 > 100000 nM T17036 C9J6LX 122191463 IC50 > 100000 nM T17036 C75NJO 122191464 IC50 > 100000 nM T17036 C50VYK 122191465 IC50 > 100000 nM T17036 CSKY20 122191466 IC50 > 100000 nM T17036 CS3L8H 122191467 IC50 = 5011.87 nM T17036 CZ2NV1 122191468 IC50 > 100000 nM T17036 CYTW93 122191469 IC50 = 79432.82 nM T17036 CZV45H 122191470 IC50 = 50118.72 nM T17036 CF6I2N 122191471 IC50 > 100000 nM T17036 CZU02B 122191472 IC50 = 25118.86 nM T17036 CE27AS 122191473 IC50 > 100000 nM T17036 CAJ28B 122191475 IC50 > 100000 nM T17036 C36PDK 122191476 IC50 > 100000 nM T17036 CQ04FW 122191477 IC50 > 100000 nM T17036 C12OHA 122191478 IC50 = 100000 nM T17036 CL2K0J 122191479 IC50 = 100000 nM T17036 CT6HG3 122191480 IC50 > 100000 nM T17036 CK7LD6 122191481 IC50 > 100000 nM T17036 CMJ72N 122191482 IC50 > 100000 nM T17036 C6H2YQ 122383780 IC50 = 5000 nM T17036 CT2UZ4 125377518 IC50 = 45000 nM T17036 CO1F4A 135567128 IC50 = 501.19 nM T17036 CE1SW8 136053677 IC50 = 501.19 nM T17036 CMW30T 136053680 IC50 = 398.11 nM T17036 C6IJ5M 136053683 IC50 = 398.11 nM T17036 CNY5T7 136053684 IC50 = 125.89 nM T17036 C2V6MX 136644692 IC50 > 100000 nM T17036 D00YEV 5281605 IC50 = 3000 nM T17036 D07IOY 10365 IC50 = 6309.57 nM T17036 D08IZY 3080614 IC50 > 100000 nM T17036 D0B2WZ 15331 IC50 > 100000 nM T17036 D0S3DD 56963315 IC50 = 19952.62 nM T17036 D0T3PW 5281672 IC50 = 3000 nM T17036 D0X5US 459617 IC50 = 200 nM T05152 D09ZZW 503536 IC50 = 1500 nM T05152 C6IQV0 482174 IC50 = 5700 nM T05152 CY61LO 487910 IC50 = 1700 nM T05152 C6K5JV 487911 IC50 = 16000 nM T05152 C3J5VH 487912 IC50 = 1000 nM T05152 CZNK70 487918 IC50 = 330 nM T05152 CDN3F2 487919 IC50 = 1630 nM T05152 CT76XW 487920 IC50 = 2100 nM T05152 CVA82G 487921 IC50 = 460 nM T05152 CBR46W 487922 IC50 = 1400 nM T05152 CAJ64Q 490750 IC50 < 1000 nM T05152 CMO49H 491114 IC50 = 4300 nM T05152 COB17R 492544 IC50 > 50000 nM T05152 C68MZE 492548 IC50 > 100000 nM T05152 C4JO9E 492549 IC50 = 3280 nM T05152 C1JEY2 492550 IC50 = 300 nM T05152 CRML27 492552 IC50 = 380 nM T05152 C84QRW 493418 IC50 = 5700 nM T05152 CY1WF7 497453 IC50 = 3000 nM T05152 C43PXV 503499 IC50 = 2400 nM T05152 C2BSI5 503516 IC50 = 14000 nM T05152 CFRT87 503517 IC50 = 5400 nM T05152 C3JB0U 503520 IC50 = 13000 nM T05152 CA72XJ 503521 IC50 = 5200 nM T05152 CF14KO 503522 IC50 = 7400 nM T05152 CH18YP 503523 IC50 = 4600 nM T05152 CG6T1D 503524 IC50 = 4100 nM T05152 CLY7T8 503525 IC50 = 750 nM T05152 C37MIA 503526 IC50 = 1000 nM T05152 C8U2AD 503527 IC50 = 12000 nM T05152 CO6R4G 503528 IC50 = 2000 nM T05152 CHA5F8 503529 IC50 > 50000 nM T05152 C41DVG 503530 IC50 = 21000 nM T05152 C5XRJ6 503531 IC50 = 1200 nM T05152 CI1V6W 503532 IC50 > 50000 nM T05152 C84DXH 503533 IC50 = 1400 nM T05152 C7R3CM 503534 IC50 = 2000 nM T05152 CCMU16 503535 IC50 = 3000 nM T05152 C1E4IO 504181 IC50 = 2700 nM T05152 CEJ6U1 504182 IC50 = 1800 nM T05152 CZDS90 504183 IC50 = 1600 nM T05152 C04ONL 504184 IC50 = 2200 nM T05152 C65XPH 504185 IC50 = 11000 nM T05152 CRZN68 504186 IC50 = 42000 nM T05152 CK8CA2 504187 IC50 > 60000 nM T05152 C01MYV 504188 IC50 = 5800 nM T05152 C4C5WD 504189 IC50 = 4300 nM T05152 CIB52E 504190 IC50 = 230 nM T05152 CQ6L1G 504191 IC50 = 12000 nM T05152 C4CW5A 504192 IC50 > 60000 nM T05152 C09ACU 504193 IC50 > 60000 nM T05152 C7T0AD 504194 IC50 = 1300 nM T05152 C7VZY1 504195 IC50 > 60000 nM T05152 CU4EK0 504196 IC50 = 3600 nM T05152 COUS53 504197 IC50 = 5300 nM T05152 CTE3B4 504198 IC50 = 7700 nM T05152 CT81MP 504676 IC50 = 3500 nM T05152 C9FI5K 504680 IC50 = 10600 nM T05152 C8IFN4 504681 IC50 = 31000 nM T05152 CV6OY3 506523 IC50 = 1400 nM T05152 CQX7S4 506524 IC50 = 390 nM T05152 CXD73I 506525 IC50 = 1800 nM T05152 C6ANI5 506528 IC50 = 9000 nM T05152 CRU30I 507613 IC50 = 900 nM T05152 CI8SQ4 511361 IC50 > 50000 nM T05152 C02LPN 511362 IC50 = 30000 nM T05152 CJIW67 511363 IC50 = 13000 nM T05152 C3KG1M 511364 IC50 = 43000 nM T05152 CU85HK 511365 IC50 = 10700 nM T05152 C20EKN 511366 IC50 = 5900 nM T05152 C3FX8J 511367 IC50 = 31000 nM T05152 C4DEY1 511368 IC50 = 3700 nM T05152 CC2J9M 511369 IC50 = 5600 nM T05152 CIU5M2 511370 IC50 = 11000 nM T05152 C5CG4I 511371 IC50 = 5000 nM T05152 CTO87P 511372 IC50 = 2700 nM T05152 C5BJ6S 511373 IC50 = 26000 nM T05152 CDWB40 511374 IC50 = 15000 nM T05152 CDH29C 511375 IC50 = 31000 nM T05152 C8ZJD7 511376 IC50 = 31000 nM T05152 CJ56OH 513150 IC50 < 10000 nM T05152 C5BN4U 513891 IC50 = 12000 nM T05152 CVI54C 657065 IC50 = 1200 nM T05152 CUC54L 3008068 IC50 = 5000 nM T05152 CJ5NO6 3008069 IC50 = 34000 nM T05152 CQO9Y3 3008070 IC50 > 32000 nM T05152 CXM1K9 3008071 IC50 > 50000 nM T05152 CJ2NY3 3008418 IC50 = 20000 nM T05152 CIJ2T0 3008419 IC50 > 50000 nM T05152 CWD1X0 3008420 IC50 = 14000 nM T05152 C4K2JP 3008421 IC50 > 50000 nM T05152 CAN83S 3008422 IC50 = 13000 nM T05152 CMDQ27 4468931 IC50 = 1800 nM T05152 CK9WY1 5278824 IC50 = 100 nM T05152 C5MEQ4 5278825 IC50 = 110 nM T05152 C1F0AN 5278826 IC50 = 45 nM T05152 CV0O6S 5482516 IC50 = 15600 nM T05152 CEM30Z 5483089 IC50 = 8900 nM T05152 CJL21S 9853197 IC50 = 60 nM T05152 CJW4M9 9917616 IC50 = 11000 nM T05152 C39ZBC 10207572 IC50 = 30000 nM T05152 CGA86Z 10259200 IC50 = 12000 nM T05152 CJ46UK 10439772 IC50 = 420 nM T05152 COM8C5 21148125 IC50 = 16000 nM T05152 C1TW3V 22209806 IC50 > 50000 nM T05152 C8GVX3 22209808 IC50 > 50000 nM T05152 C6AS7E 22209811 IC50 = 3300 nM T05152 CLW13P 22209812 IC50 = 1700 nM T05152 C1TA6Z 22209813 IC50 = 440 nM T05152 CGUC83 22210989 IC50 = 58000 nM T05152 CV97ER 22210996 IC50 = 18000 nM T05152 C2BA1K 22211000 IC50 = 27000 nM T05152 C78AKX 22211010 IC50 > 100000 nM T05152 CL7M9B 22211011 IC50 = 32000 nM T05152 C1L8TE 22211012 IC50 = 18000 nM T05152 C0NYS5 22211016 IC50 = 50000 nM T05152 C67QJW 22211018 IC50 > 100000 nM T05152 CV9S2O 22211019 IC50 = 13000 nM T05152 C4UB6Q 22211020 IC50 = 14000 nM T05152 CBUV46 22211021 IC50 = 62000 nM T05152 CS9B7N 22211022 IC50 > 100000 nM T05152 CK81WO 25078062 IC50 = 3400 nM T05152 CYDW71 44268661 IC50 > 60000 nM T05152 C6S3AT 44268682 IC50 > 60000 nM T05152 CDJ0X4 44308299 IC50 > 100000 nM T05152 CIO1C2 44308345 IC50 > 100000 nM T05152 CX14BI 44308422 IC50 > 100000 nM T05152 CE3PS8 44308752 IC50 = 34000 nM T05152 CK2P5O 44375061 IC50 > 50000 nM T05152 C4CVW1 44375110 IC50 > 50000 nM T05152 C72KUL 44375154 IC50 = 9400 nM T05152 C1SBO9 44375192 IC50 > 50000 nM T05152 C42GUE 44375229 IC50 = 5300 nM T05152 CX76FI 44388198 IC50 = 350 nM T05152 CVW6O4 44399745 IC50 = 79432.82 nM T05152 CDRP83 44399750 IC50 = 50118.72 nM T05152 CW6NY8 44399751 IC50 = 5011.87 nM T05152 CM5W8Q 44399752 IC50 = 6309.57 nM T05152 C34WSP 44399753 IC50 = 10000 nM T05152 CE0T1O 44399754 IC50 = 1995.26 nM T05152 CT86CR 44399784 IC50 = 25118.86 nM T05152 C6GWS9 44399837 IC50 = 31622.78 nM T05152 C4AI1T 44399861 IC50 = 100000 nM T05152 CTX79F 44399866 IC50 = 25118.86 nM T05152 CP4KB7 44399867 IC50 = 794.33 nM T05152 C0WRU5 44399868 IC50 = 15848.93 nM T05152 C8JP2A 44399889 IC50 = 50118.72 nM T05152 CO4H3V 44399938 IC50 = 10000 nM T05152 CYH7F9 44399975 IC50 = 6309.57 nM T05152 CZRF38 44399976 IC50 = 6309.57 nM T05152 CATH48 44399977 IC50 = 6309.57 nM T05152 CL9NS3 44399978 IC50 > 199526.23 nM T05152 C9YO4K 44399979 IC50 > 199526.23 nM T05152 CX8M3O 44400003 IC50 = 39810.72 nM T05152 C4X1OG 44400004 IC50 = 19952.62 nM T05152 C5EV1S 44400005 IC50 = 158489.32 nM T05152 CFRU27 44400006 IC50 = 199526.23 nM T05152 C7FO3T 44400007 IC50 = 251188.64 nM T05152 CA6P2U 44400008 IC50 = 100000 nM T05152 CQP47M 44400009 IC50 = 7943.28 nM T05152 CCRB97 44400010 IC50 = 3981.07 nM T05152 CT40SR 44400033 IC50 = 31622.78 nM T05152 CA96HO 44400076 IC50 > 1000000 nM T05152 CX7O2Z 44400112 IC50 > 199526.23 nM T05152 C6Z5NC 44400113 IC50 > 199526.23 nM T05152 C6PCE5 44400114 IC50 = 31622.78 nM T05152 C95CRD 44400115 IC50 = 19952.62 nM T05152 CW5G3Z 73347065 IC50 > 50000 nM T05152 C6TNQ8 135412361 IC50 = 800 nM T05152 C53AWL 135434400 IC50 = 100 nM T74073 C7DO2P 70981589 IC50 = 2668 nM T74073 C0WC3B 70981821 IC50 = 1761 nM T74073 C23ARZ 70982089 IC50 = 1536 nM T74073 CNKX61 70982376 IC50 = 602 nM T74073 CH7J2X 70982568 IC50 = 28 nM T74073 CM4T3D 70983036 IC50 = 2982 nM T74073 C97WBL 70983181 IC50 = 212 nM T74073 C61DAP 70983443 IC50 = 45 nM T74073 C9ASG6 70984064 IC50 = 403 nM T74073 CVT09B 71007225 IC50 = 4807 nM T74073 C1BND0 71007226 IC50 = 983 nM T74073 C35VQT 71007233 IC50 = 620 nM T74073 C0O7XS 71007248 IC50 = 286 nM T74073 CWK3P9 71007275 IC50 = 5120 nM T74073 CT23JC 71007294 IC50 = 2530 nM T74073 C34ANW 71007298 IC50 = 221 nM T74073 CILG13 71007335 IC50 = 5007 nM T74073 C2K6EB 71007339 IC50 = 1760 nM T74073 CZ1TG7 71007340 IC50 = 522 nM T74073 CR1G6M 71007342 IC50 = 3440 nM T74073 C0KEC3 71007349 IC50 = 6599 nM T74073 CBF2N4 71007352 IC50 > 15800 nM T74073 CO3C5Z 71007358 IC50 = 6100 nM T74073 C8Y3VW 71465328 IC50 = 258 nM T74073 CGY4Z5 71730239 IC50 = 78 nM T74073 CS2RT7 71730241 IC50 = 30 nM T74073 CEZ0Y3 71730242 IC50 = 65 nM T74073 CR80EU 71730367 IC50 = 44 nM T74073 C09BGX 71731146 IC50 = 110 nM T74073 C5ES1L 71731394 IC50 = 184 nM T74073 CC2UI1 71731515 IC50 = 23 nM T74073 C87XSZ 71731781 IC50 = 29 nM T74073 C8VPO2 71731919 IC50 = 1635 nM T74073 CVF34X 73056835 IC50 = 25 nM T74073 CVY2Z3 73056836 IC50 = 40 nM T74073 C25CJV 73057145 IC50 = 14 nM T74073 CI57QV 89782019 IC50 = 31 nM T74073 CH8JN1 89783250 IC50 = 148 nM T74073 C1CL8I 89783341 IC50 = 26 nM T74073 CUNJ79 89783434 IC50 = 22 nM T74073 C2K3DA 89783801 IC50 = 11 nM T74073 CPQ9L3 89783993 IC50 = 143 nM T74073 C16ZQO 89784003 IC50 = 407 nM T74073 CX2H4B 89784954 IC50 = 4560 nM T74073 C0JIS8 89793954 IC50 = 5760 nM T74073 CXF3T0 90058666 IC50 = 16 nM T74073 C1UJ8Q 90058675 IC50 = 100 nM T74073 CWRJ32 90058676 IC50 = 106 nM T74073 CYZ98S 90058679 IC50 = 26 nM T74073 CFH4L6 90058683 IC50 = 20 nM T74073 CV9KG7 90058690 IC50 = 20 nM T74073 CP13IU 90058693 IC50 = 880 nM T74073 C56AJL 90058786 IC50 = 370 nM T74073 C35WJR 90058791 IC50 = 21 nM T74073 CCA78J 90058814 IC50 = 37 nM T74073 CN6H2I 90058905 IC50 = 25 nM T74073 C7DVW3 90058906 IC50 = 37 nM T74073 C75FLG 90326903 IC50 = 49 nM T74073 CN0V6L 90326906 IC50 = 142 nM T74073 C1W4DO 134135721 IC50 = 115 nM T74073 CX3A0W 134146922 IC50 = 31 nM T74073 CU35GB 155517528 EC50 = 90 nM T74073 CY49NZ 155518625 EC50 = 93 nM T74073 CO58XZ 155519799 EC50 = 18 nM T74073 CY7EM6 155525492 EC50 = 33 nM T74073 CX59UT 155526046 EC50 = 98 nM T74073 CS9W1N 155531462 EC50 = 59 nM T74073 CY59IV 155531989 EC50 = 70 nM T74073 CL7U8D 155534608 EC50 = 37 nM T74073 C68KHN 155539424 IC50 = 2870 nM T74073 CWQ7F0 155541490 EC50 = 69 nM T74073 C2IG7U 155543022 IC50 > 2000 nM T74073 CRG0K4 155544306 IC50 = 1380 nM T74073 CPB87M 155545130 EC50 = 53 nM T74073 CNL4B8 155546196 IC50 = 1642 nM T74073 CC83QJ 155547453 EC50 = 133 nM T74073 CEDN41 155550408 EC50 = 27 nM T74073 CB73CQ 155551312 EC50 = 61 nM T74073 CG26ND 155552144 IC50 = 1142 nM T74073 C62DJU 155558058 IC50 = 5960 nM T74073 CM0UH7 155559265 EC50 = 128 nM T74073 CRLP86 155560079 EC50 = 28 nM T74073 CJ9M3Y 155563039 IC50 = 88 nM T74073 C43CBF 155566090 EC50 = 51 nM T74073 C9WB2L 155566373 EC50 = 36 nM T74073 C1B7YH 155566566 IC50 = 127 nM T74073 C04THL 155567360 EC50 = 32 nM T74073 C4ED0G 155568443 IC50 = 167 nM T74073 CV8W5R 155569485 EC50 = 13 nM T15848 D09KTS 24821094 IC50 = 0.5 nM T15848 D0E6XR 3062316 IC50 = 297 nM T15848 D0OB0F 5328940 IC50 = 282 nM T15848 D02TUL 118115473 IC50 = 592 nM T15848 D04BFC 59174488 IC50 = 6.2 nM T15848 D08AOZ 86582336 IC50 = 10 nM T15848 D0E3TC 44259 IC50 = 43.1 nM T15848 D0G5XV 135565884 IC50 = 2 nM T15848 D0QX8X 71479709 IC50 = 37.9 nM T15848 C9F1AO 24821023 IC50 = 78 nM T15848 CSNC57 25110758 IC50 > 10000 nM T15848 C0GOX5 25110759 IC50 > 10000 nM T15848 CC2R7S 25110760 IC50 > 10000 nM T15848 CA98KR 44432441 IC50 = 22000 nM T15848 C3VRO9 44557921 IC50 > 10000 nM T15848 C8ZRE3 53356518 IC50 = 14 nM T15848 CJBL48 56925034 IC50 = 116 nM T15848 CV13QY 58540422 IC50 = 230 nM T15848 CT3EW2 59292007 IC50 > 1000 nM T15848 CZ3TG1 59375154 IC50 = 162 nM T15848 CV63UL 67240318 IC50 > 10000 nM T15848 C7VJ6A 70647728 IC50 = 13 nM T15848 COU73Y 71226944 IC50 = 63 nM T15848 C40JOZ 71235465 IC50 = 232 nM T15848 CZM1K4 71765510 IC50 = 57 nM T15848 C5MJ0H 71765626 IC50 = 57 nM T15848 C9OQ2I 72710839 IC50 > 10000 nM T15848 CX75YR 73352604 IC50 = 251.19 nM T15848 CSG38E 89455222 IC50 = 5.3 nM T15848 C37DUM 121293882 IC50 = 6.4 nM T15848 CXQR89 121294143 IC50 = 0.9 nM T15848 CFKD32 122191637 IC50 = 41 nM T15848 CLM7K3 122604539 IC50 > 10000 nM T15848 C01JHI 122604566 IC50 > 10000 nM T15848 CGFK71 130429248 IC50 = 306.45 nM T15848 CV89JM 132231876 IC50 = 2.3 nM T15848 C59HOQ 134277578 IC50 = 1.78 nM T15848 C0PZ5R 134277599 IC50 = 2.27 nM T15848 C7PWJ2 134277617 IC50 = 0.09 nM T15848 CRA2H1 134277633 IC50 = 4.32 nM T15848 CXJ8I0 134277643 IC50 = 1.65 nM T15848 C02RIA 134277647 IC50 = 0.2 nM T15848 CGH42R 134277652 IC50 = 0.67 nM T15848 COA14U 134277654 IC50 = 0.16 nM T15848 CQK0B5 134277685 IC50 = 4.5 nM T15848 C6S8VC 134277696 IC50 = 2 nM T15848 C49PIO 134277748 IC50 = 3.13 nM T15848 CD7VK4 134277767 IC50 = 3.16 nM T15848 CZ5E6L 134277773 IC50 = 1.96 nM T15848 C2CFK7 134277780 IC50 = 0.98 nM T15848 C6E7LW 134277790 IC50 = 0.62 nM T15848 C6T7NW 134277796 IC50 = 0.1 nM T15848 CU8ZP5 134277800 IC50 = 0.74 nM T15848 CTR4K6 134277828 IC50 = 0.11 nM T15848 C3Z4AT 137321159 IC50 > 10000 nM T15848 CZOD53 137633880 IC50 = 378 nM T15848 C7BJY5 137636807 IC50 = 191 nM T15848 CO89DX 137649100 IC50 = 170 nM T15848 CINE03 137652514 IC50 = 428 nM T15848 C28QUP 137652864 IC50 = 114.8 nM T15848 CRWA29 139030520 IC50 = 227 nM T15848 C9ZYG8 141366083 IC50 = 56 nM T15848 C4OD9Q 145967187 IC50 = 1.4 nM T15848 CE31VG 145979714 IC50 > 10000 nM T15848 C9BX4U 145988956 IC50 = 8960 nM T15848 C3NA2I 155519537 IC50 = 44 nM T15848 D01RHR 71519693 IC50 = 8.2 nM T15848 D04PEI 11467730 IC50 = 17000 nM T15848 D06BJG 71556703 IC50 = 6.3 nM T15848 D0N0LN 46908026 IC50 = 64 nM T24595 C62ATV 1718 IC50 = 8 nM T24595 CM92QV 4427 IC50 = 142600000 nM T24595 CV1Y8U 33346 IC50 = 2410 nM T24595 CIF84X 55903 IC50 = 9.3 nM T24595 C0NI8J 55905 IC50 = 19.8 nM T24595 CWO60H 55906 IC50 = 12.9 nM T24595 CP5XV0 55907 IC50 = 13.7 nM T24595 C4O3YG 55908 IC50 = 99.7 nM T24595 CQC2Y8 73094 IC50 = 142600000 nM T24595 C8TX4U 403858 IC50 = 2500000 nM T24595 CS65PQ 3015798 IC50 = 5.6 nM T24595 C8H7TV 5172643 IC50 = 2060000 nM T24595 CWK94T 12241396 IC50 = 2300000 nM T24595 C4MTL2 12925726 IC50 = 6.6 nM T24595 C7PNY5 12925730 IC50 = 16.3 nM T24595 CW4EJ0 12925742 IC50 = 17.6 nM T24595 C4SJ8H 13245401 IC50 = 0.67 nM T24595 CDG80P 13245402 IC50 = 300 nM T24595 CV9UK1 13590035 IC50 = 5.4 nM T24595 CA26FM 14480651 IC50 = 27.3 nM T24595 CIB7M6 14480685 IC50 = 38.5 nM T24595 CZ92FX 16728293 IC50 = 390000 nM T24595 CH5BJ6 19508766 IC50 = 90000 nM T24595 C9VMK3 43392945 IC50 = 2800000 nM T24595 CU97QY 43417711 IC50 = 540000 nM T24595 CD2OX4 43418370 IC50 = 60000 nM T24595 C4ILD3 43418690 IC50 = 3000000 nM T24595 CN3TD7 44365378 IC50 = 33 nM T24595 CSN3E7 44365380 IC50 = 11.4 nM T24595 CY5ZU1 44365482 IC50 = 7.2 nM T24595 CW86PH 44365662 IC50 = 28.5 nM T24595 C3PVW9 53484097 IC50 = 110000 nM T24595 CKV76T 53484116 IC50 = 440000 nM T24595 CDQ63K 56657915 IC50 = 17000000 nM T24595 CVK51J 56657916 IC50 = 5760000 nM T24595 C56YJP 56657917 IC50 = 9250000 nM T24595 C2UIA7 56664885 IC50 = 8000000 nM T24595 CKTN91 56665089 IC50 = 3980000 nM T24595 C10WLM 56665090 IC50 = 2400000 nM T24595 CS64UK 56665091 IC50 = 3310000 nM T24595 CSQ1U7 56668303 IC50 = 72000000 nM T24595 CNX79C 56668304 IC50 = 7900000 nM T24595 CKZ7L3 56671784 IC50 = 23000000 nM T24595 CG9K5O 56671785 IC50 = 17400000 nM T24595 CWQ38L 56672041 IC50 = 800000 nM T24595 CJ9Y3T 56672042 IC50 = 470000 nM T24595 CJ7R0Y 56675194 IC50 = 14000000 nM T24595 CW69FO 56675418 IC50 = 34600000 nM T24595 CM7K0F 56678493 IC50 = 32000 nM T24595 CU4XC9 56678768 IC50 = 4800000 nM T24595 C89QCV 56682077 IC50 = 2400000 nM T24595 CN3DG9 56682078 IC50 = 3310000 nM T24595 CTR3Y1 56682079 IC50 = 3300000 nM T24595 CYN52A 56930433 IC50 = 210000 nM T24595 CSM6V7 57390307 IC50 = 2210000 nM T24595 C6XEZ2 57390964 IC50 = 3840000 nM T24595 CFLN09 57390965 IC50 = 9580000 nM T24595 CV1Y2I 57390966 IC50 = 2990000 nM T24595 CLS1T6 57392743 IC50 = 7110000 nM T24595 CZV10B 57392744 IC50 = 7050000 nM T24595 C6YD8A 57392745 IC50 = 9900000 nM T24595 CDN2U4 57392746 IC50 = 4980000 nM T24595 C5GW7Y 57394476 IC50 = 3800000 nM T24595 CX7CJ4 57394477 IC50 = 7630000 nM T24595 CE2H9J 57394478 IC50 = 130000 nM T24595 CYG16N 57394479 IC50 = 1580000 nM T24595 CM9G8X 57394480 IC50 = 9300000 nM T24595 C4UPY5 57394481 IC50 = 3310000 nM T24595 CP5Z4I 57394482 IC50 = 8980000 nM T24595 CK8BO3 57394483 IC50 = 9350000 nM T24595 C29RSE 57396240 IC50 = 5960000 nM T24595 CU27KZ 57396241 IC50 = 2510000 nM T24595 C4BH1T 57396242 IC50 = 9300000 nM T24595 CW04QS 57398034 IC50 = 6300000 nM T24595 CS2K6I 57398035 IC50 = 9000000 nM T24595 CDF68T 57398036 IC50 = 9500000 nM T24595 C3IVH7 57398037 IC50 = 8920000 nM T24595 C2ANG1 57399695 IC50 = 7000000 nM T24595 CZ6W5G 57399696 IC50 = 7180000 nM T24595 C1PU3X 57399697 IC50 = 9840000 nM T24595 CENZ91 57401454 IC50 = 2450000 nM T24595 C6O5MP 57401455 IC50 = 2350000 nM T24595 C1ECW9 57401456 IC50 = 4200000 nM T24595 C9YE0K 57403193 IC50 = 5630000 nM T24595 C8KV6C 57403194 IC50 = 7410000 nM T24595 CJ2D0T 60142639 IC50 = 140000 nM T24595 CG97OL 60142640 IC50 = 60000 nM T24595 CC9YO7 60142777 IC50 = 460000 nM T24595 CANP75 60142778 IC50 = 380000 nM T24595 CM2F5K 61236018 IC50 = 1700000 nM T24595 C4OMA3 70683428 IC50 = 5750000 nM T24595 CXC26K 70683504 IC50 = 63000 nM T24595 CM5U8J 70685601 IC50 = 10700000 nM T24595 C8EHG4 70685602 IC50 = 1550000 nM T24595 C4EAF7 70685603 IC50 = 1590000 nM T24595 C2IJ9T 70685604 IC50 = 8420000 nM T24595 C8JD6P 70687753 IC50 = 3180000 nM T24595 C5QD3B 70687754 IC50 = 11500000 nM T24595 CJ6R2C 70687755 IC50 = 470000 nM T24595 CJQ53M 70687756 IC50 = 1800000 nM T24595 C68XIT 70689735 IC50 = 8860000 nM T24595 CS2YR0 70689736 IC50 = 310000 nM T24595 C1BH0M 70689804 IC50 = 7500000 nM T24595 CED0G6 70691883 IC50 = 2400000 nM T24595 C16VNO 70691884 IC50 = 7520000 nM T24595 C6YI0Q 70691885 IC50 = 4020000 nM T24595 CSA91L 70691886 IC50 = 3290000 nM T24595 CRU79W 70691944 IC50 = 1770000 nM T24595 C0NTP6 70693921 IC50 = 1640000 nM T24595 C1ND4S 70693922 IC50 = 1270000 nM T24595 C0FHM8 70693994 IC50 = 5060000 nM T24595 C1J4SK 70693995 IC50 = 1030000 nM T24595 CO32UN 70693996 IC50 = 1810000 nM T24595 C0TBN2 70696118 IC50 = 1250000 nM T24595 C2YNO8 71569407 IC50 = 80000 nM T24595 CGF34J 71569408 IC50 = 7320000 nM T24595 C5PNQ6 71569409 IC50 = 2450000 nM T24595 C6FE4D 71569410 IC50 = 340000 nM T24595 CKX18T 71569568 IC50 = 6040000 nM T24595 CJ5O4S 71569569 IC50 = 5450000 nM T24595 C56MFY 71569570 IC50 = 280000 nM T24595 CWT3P4 71569571 IC50 = 1060000 nM T24595 C5SW3D 71569572 IC50 = 1620000 nM T24595 CI8A2S 71569573 IC50 = 1090000 nM T24595 C0IDP1 71569574 IC50 = 540000 nM T24595 CJ0UK5 71569740 IC50 = 5080000 nM T24595 CZ1PQ7 71569741 IC50 = 410000 nM T24595 C37GHZ 71569742 IC50 = 5730000 nM T24595 CHG2T1 71569743 IC50 = 1430000 nM T24595 CMBJ16 71569744 IC50 = 8920000 nM T24595 C6HVQ5 71569745 IC50 = 3240000 nM T24595 CFLB03 71569746 IC50 = 3780000 nM T24595 CP7Q1J 71713187 IC50 = 6020000 nM T24595 CWFT30 71713188 IC50 = 2700000 nM T24595 CVJ24O 71713189 IC50 = 5600000 nM T24595 C6DQ8P 71713190 IC50 = 3070000 nM T24595 CRU7F0 71713191 IC50 = 2950000 nM T24595 C2V6JM 71713192 IC50 = 1210000 nM T24595 C1OXE2 71713193 IC50 = 2000000 nM T24595 CH2W0I 71713194 IC50 = 1875000 nM T24595 CG8PM9 71713342 IC50 = 2070000 nM T24595 C6P1TG 71713343 IC50 = 5220000 nM T24595 CH8UN6 71713344 IC50 = 760000 nM T24595 C21PDW 71713345 IC50 = 2400000 nM T24595 CC1M4X 71713346 IC50 = 780000 nM T24595 C74JNL 71713347 IC50 = 1830000 nM T24595 C93WVU 71713348 IC50 = 790000 nM T24595 CSQW49 71713349 IC50 = 9100000 nM T24595 CXUM74 71713481 IC50 = 760000 nM T24595 C8DZR1 71713482 IC50 = 530000 nM T24595 C8RU2O 71713483 IC50 = 1520000 nM T24595 C08TSP 71713484 IC50 = 380000 nM T24595 CTG81I 71713485 IC50 = 330000 nM T24595 C6E0CD 71713486 IC50 = 880000 nM T24595 CMQ6N3 71713487 IC50 = 10000000 nM T24595 C7YFA9 71713626 IC50 = 10000 nM T24595 CH1EW8 71713627 IC50 = 940000 nM T24595 CZ0GO3 71717981 IC50 = 2780000 nM T24595 C1BNM3 86567056 IC50 = 26770 nM T24595 C6FL8Z 90468998 IC50 = 1400 nM T24595 CW5JT8 90644232 IC50 = 240000 nM T24595 C9UR5K 90644233 IC50 > 100000 nM T24595 CW17IT 90644234 IC50 > 100000 nM T24595 CCXV81 90644235 IC50 = 24600 nM T24595 CEMY61 90644236 IC50 = 21400 nM T24595 CFC6J3 90644237 IC50 = 2300 nM T24595 CL13ZU 90644238 IC50 = 9300 nM T24595 C72SAW 90644239 IC50 = 7800 nM T24595 C7WQ0L 90644240 IC50 = 10100 nM T24595 CJR78O 90644241 IC50 = 5700 nM T24595 CA42XM 90644242 IC50 = 25400 nM T24595 CFU8J5 90644243 IC50 = 12100 nM T24595 C5BF2R 90644244 IC50 = 14400 nM T24595 COR0G5 90644245 IC50 = 14400 nM T24595 CGS6B5 90644246 IC50 = 6400 nM T24595 C0IAS7 90644247 IC50 = 20300 nM T24595 CDO4Q3 90644248 IC50 = 26800 nM T24595 CCZ59D 90644249 IC50 = 8400 nM T24595 CF17LQ 90644250 IC50 = 6600 nM T24595 C8UZW0 90644251 IC50 = 27900 nM T24595 C9ZMO6 90644252 IC50 = 29900 nM T24595 CMN82Z 90644253 IC50 = 9400 nM T24595 CU24TA 90644254 IC50 = 23900 nM T24595 CN7HR6 90644255 IC50 = 11500 nM T24595 C4QLS0 90644256 IC50 = 20500 nM T24595 CR6U8C 122182848 IC50 = 15140 nM T24595 CN05MJ 122182849 IC50 = 2380 nM T24595 CCY4R1 122182850 IC50 = 1260 nM T24595 CR56NU 122182851 IC50 = 9430 nM T24595 C1BC6L 122182852 IC50 = 11320 nM T24595 CLX57F 122182853 IC50 = 17740 nM T24595 CZY8S4 122182854 IC50 = 16130 nM T24595 C0NY8C 122182855 IC50 = 5730 nM T24595 CH4MP7 122182856 IC50 = 25430 nM T24595 C9J6AP 122182857 IC50 = 10860 nM T24595 C6A1SN 122182858 IC50 = 9460 nM T24595 CUK31Q 122182859 IC50 = 23870 nM T24595 C2CZ0Y 122182860 IC50 = 24530 nM T24595 CM12RO 122182861 IC50 = 8450 nM T24595 CUY04Z 122182862 IC50 = 23740 nM T24595 C4HCB6 122182863 IC50 = 7470 nM T24595 C2C9XB 122182864 IC50 = 25910 nM T24595 CK5TF1 122182865 IC50 = 13110 nM T24595 C26CPD 122182866 IC50 = 24380 nM T24595 C56CUE 122182867 IC50 = 5870 nM T24595 CZL6D5 122182868 IC50 = 4320 nM T24595 CE5D1S 122182870 IC50 = 3440 nM T24595 CY7FE8 122182871 IC50 = 28330 nM T24595 CZQV71 122182872 IC50 = 2420 nM T24595 C83BPN 122182873 IC50 = 16550 nM T24595 CGYC30 122182874 IC50 > 100000 nM T24595 CQ1PF9 122182876 IC50 > 100000 nM T24595 D0F9YV 44365677 IC50 = 3.3 nM T03385 C4CX0W 619958 IC50 = 23000 nM T03385 CS29HL 715103 IC50 = 18600 nM T03385 CAS07I 715106 IC50 > 30000 nM T03385 C13UKR 829570 IC50 = 10700 nM T03385 CH1C3S 1130426 IC50 = 9800 nM T03385 CES28Q 1889993 IC50 = 10000 nM T03385 CKZE78 5306660 IC50 = 12400 nM T03385 C7MPE6 7680155 IC50 = 10200 nM T03385 CF81QM 8057056 IC50 = 3200 nM T03385 CRO0V4 8057213 IC50 = 13000 nM T03385 C7CUA4 19591131 IC50 = 14700 nM T03385 CRV56W 25012734 IC50 = 7700 nM T03385 CYQW64 25012735 IC50 = 9600 nM T03385 CYT7H9 25012739 IC50 = 8600 nM T03385 C7P2RK 25012896 IC50 = 2800 nM T03385 CPZ9O0 25012897 IC50 = 7100 nM T03385 C3IKD2 25012898 IC50 = 1000 nM T03385 CZC52F 25012899 IC50 = 3000 nM T03385 C7QHW6 25012900 IC50 = 4900 nM T03385 C6OZB1 25013058 IC50 = 9500 nM T03385 CEGS28 25013059 IC50 = 14400 nM T03385 C6LMU3 25013390 IC50 = 6800 nM T03385 C50QTU 25013393 IC50 = 1900 nM T03385 C2Z1PR 25013555 IC50 = 2300 nM T03385 CB96AF 25013557 IC50 = 900 nM T03385 C3J6DU 50991753 IC50 = 17000 nM T03385 C90VTC 53363650 IC50 > 30000 nM T03385 D06OVX 65094 IC50 = 300 nM T99340 D05ROI 44462760 IC50 = 53200 nM T99340 D0H0EQ 24826799 IC50 = 12 nM T99340 D0W5HK 216239 IC50 = 1500 nM T99340 D02XNW 5494449 IC50 = 208 nM T99340 D0LQ3L 77108121 IC50 = 0.4 nM T99340 C09BCS 23578 Ki = 63.1 nM T99340 C76XNU 643953 IC50 = 754 nM T99340 C5IOS0 670041 EC50 = 4100 nM T99340 C7X5WE 2828334 EC50 = 182 nM T99340 C86MXJ 3063662 IC50 = 794 nM T99340 CDLJ02 3078467 IC50 = 2000 nM T99340 C8B3WY 3078469 IC50 = 2000 nM T99340 CMV76B 3078470 IC50 = 10 nM T99340 CYE04H 3078480 IC50 = 1.6 nM T99340 CZ4WV2 3670283 IC50 = 126 nM T99340 CA82YG 4628569 EC50 > 10000 nM T99340 CL70MG 4634732 EC50 = 457 nM T99340 C7TA9J 10113568 Ki = 2.042 nM T99340 CIV15Q 10113978 IC50 = 873 nM T99340 CFB81R 10317604 IC50 = 160 nM T99340 CF8Q2B 11288934 EC50 = 18 nM T99340 C8ET0Q 12791776 IC50 > 10000 nM T99340 CD2E5U 13142332 EC50 > 10000 nM T99340 C4V0BX 20895670 IC50 = 79 nM T99340 C25UKC 21081761 IC50 = 1500 nM T99340 CSFK63 23646936 IC50 = 32 nM T99340 CJ5H1Z 23646938 IC50 = 10 nM T99340 CIP7T2 23646939 IC50 = 2500 nM T99340 CI32JB 23646942 IC50 = 100 nM T99340 CX30ZW 25023828 IC50 = 73.6 nM T99340 C38PUJ 45271185 IC50 = 600 nM T99340 CS9T8F 53466952 IC50 = 61 nM T99340 C0HY3M 53467389 IC50 = 58 nM T99340 CLP04A 53467390 IC50 = 14 nM T99340 CV7C0D 53469060 IC50 = 69 nM T99340 CY04AP 53469630 IC50 = 56 nM T99340 CU4B0V 53469825 IC50 = 116 nM T99340 C5B4NV 55157876 EC50 = 1077 nM T99340 CKFP29 57971132 IC50 = 13 nM T99340 CUB9N0 60236671 EC50 = 378 nM T99340 CD8AV0 60698388 IC50 > 10000 nM T99340 CXIQ15 60723604 IC50 = 316 nM T99340 CVY1Z2 62679367 EC50 > 10000 nM T99340 CX30KT 62679368 EC50 = 8562 nM T99340 COQ08Y 62679370 EC50 = 1233 nM T99340 C9DYZ5 71816195 IC50 = 630 nM T99340 CY8O3K 72724969 IC50 = 20 nM T99340 CW7YD6 72725026 IC50 = 16 nM T99340 C5SQ7I 72725027 IC50 = 32 nM T99340 CFB69C 72725028 IC50 = 10 nM T99340 CE7G9T 72725029 IC50 = 4 nM T99340 CFR80L 72725083 IC50 = 160 nM T99340 COP05E 76310255 IC50 = 10 nM T99340 CHB93K 76313942 IC50 = 200 nM T99340 CCS63Z 76317480 IC50 = 40 nM T99340 CL0BO7 76317481 IC50 = 320 nM T99340 CFYP81 76317482 IC50 = 32 nM T99340 CFX5S0 76321210 IC50 = 4000 nM T99340 C7SD8Z 76321211 IC50 = 500 nM T99340 CKD2R6 76321212 IC50 = 63 nM T99340 C9X6CZ 76321213 IC50 = 160 nM T99340 C1EMH2 76321214 IC50 = 10 nM T99340 CW95IP 76324828 IC50 = 160 nM T99340 C35VHG 76328382 IC50 = 320 nM T99340 CUB91G 76328383 IC50 = 10 nM T99340 CAD50N 76328384 IC50 = 16 nM T99340 C4MT3A 76332057 IC50 = 25 nM T99340 C9IC1L 76332058 IC50 = 3200 nM T99340 C0K5MP 76332059 IC50 = 6.3 nM T99340 CO7J2V 76332061 IC50 = 16 nM T99340 CE09XW 76335674 IC50 = 200 nM T99340 CPUD78 77230897 IC50 = 1030 nM T99340 CB5H7C 82244347 IC50 > 10000 nM T99340 CC0US3 90345286 IC50 = 7.9 nM T99340 CM73SR 90345378 IC50 = 0.94 nM T99340 CNTP05 90345427 IC50 = 50 nM T99340 CS43ZG 90351311 Ki = 0.8 nM T99340 CR9ZV7 90351952 IC50 = 0.5 nM T99340 C4LT3Y 91885439 IC50 = 8.6 nM T99340 C28GLZ 110728326 IC50 > 1000 nM T99340 CF20OX 118557066 IC50 = 5 nM T99340 C6V5XY 118557110 IC50 = 0.4 nM T99340 C5ZQ4I 118557139 IC50 = 0.79 nM T99340 C78DEX 118557145 IC50 = 1600 nM T99340 C98CAG 118557162 IC50 = 0.4 nM T99340 CFJ27P 118557220 IC50 = 400 nM T99340 CSJR15 118557245 IC50 = 79 nM T99340 C21IGS 118557254 IC50 = 320 nM T99340 C3LR2H 118557293 IC50 = 1.6 nM T99340 CCYI79 118557322 IC50 = 0.79 nM T99340 CSD2H6 118557338 IC50 = 3.2 nM T99340 C5O4ZV 118557362 IC50 = 0.079 nM T99340 C6S0NT 118557462 IC50 = 63 nM T99340 CE8J7H 118557468 IC50 = 25 nM T99340 C02OGI 118557491 IC50 = 1 nM T99340 C42EMA 118557502 IC50 = 0.5 nM T99340 C12PXU 118557507 IC50 = 0.5 nM T99340 CS6JK9 118557559 IC50 = 794 nM T99340 CU7I5M 118564393 IC50 = 200 nM T99340 C2U3FR 118564396 IC50 = 32 nM T99340 CU0DW4 118564398 IC50 = 5 nM T99340 C7TBH3 118564402 IC50 = 0.32 nM T99340 C3KNZ5 121439991 EC50 = 28 nM T99340 CCX27F 121440014 EC50 = 74 nM T99340 CUR74H 121440015 EC50 > 3000 nM T99340 CH3CO4 121440032 EC50 = 262 nM T99340 CE0QC9 121440033 EC50 = 49 nM T99340 CJ0A5S 121440051 EC50 = 64 nM T99340 CLJI17 121446658 EC50 = 628 nM T99340 CY5A1S 121446659 EC50 = 125 nM T99340 C0HFX3 121446661 EC50 > 10000 nM T99340 C04IQZ 121446667 EC50 > 3000 nM T99340 C19DEL 121446676 EC50 = 490 nM T99340 C4FAO7 121446682 EC50 = 1234 nM T99340 CKUM01 121446684 EC50 = 56 nM T99340 CTM6K0 121446695 EC50 > 3000 nM T99340 CY61UA 121446710 EC50 = 1526 nM T99340 CWN4T7 121446721 EC50 = 1735 nM T99340 C0ZE8M 121446729 EC50 > 10000 nM T99340 CTXO48 121446730 EC50 = 898 nM T99340 C57TND 121446732 EC50 = 1254 nM T99340 CQH48Z 121446733 EC50 > 10000 nM T99340 CYTZ27 121446735 EC50 > 10000 nM T99340 C1ENL2 121446737 EC50 > 10000 nM T99340 CH68FX 121446738 EC50 = 221 nM T99340 C8SK7Y 121446739 EC50 = 628 nM T99340 C54DCI 121446741 EC50 > 10000 nM T99340 C1K5ZD 121446742 EC50 > 5000 nM T99340 CO32FQ 121446750 EC50 > 10000 nM T99340 C1FU2G 121446752 EC50 > 10000 nM T99340 CJ08HW 121446757 EC50 = 627 nM T99340 CX06JV 121446760 EC50 = 2527 nM T99340 C2ZF7V 121446761 EC50 = 8237 nM T99340 CB3I0L 121446764 EC50 = 656 nM T99340 C1H3VY 121446771 EC50 = 1308 nM T99340 C0B1WO 121446775 EC50 = 198 nM T99340 CU92HQ 121446778 EC50 = 58 nM T99340 C08KJZ 121446782 EC50 = 72 nM T99340 CVM06Q 121446783 EC50 = 36 nM T99340 CCD94Y 121446786 EC50 > 10000 nM T99340 CT8K2N 121446791 EC50 > 10000 nM T99340 C4NT5D 121446843 EC50 > 3000 nM T99340 CGP13F 121446847 EC50 = 12 nM T99340 CNH04D 121446878 EC50 = 98 nM T99340 C4QV9N 121446902 EC50 = 815 nM T99340 C8P4AE 122703561 IC50 = 10 nM T99340 C9E5DT 122703570 IC50 = 2 nM T99340 CM7C5F 122703576 IC50 = 7.9 nM T99340 CF5WY1 122703578 IC50 = 10 nM T99340 CF4PR9 122703579 IC50 = 16 nM T99340 C74SQF 122703581 IC50 = 13 nM T99340 CPA2Z5 122703584 IC50 = 10 nM T99340 CW70QA 122703585 IC50 = 63 nM T99340 CA6Z5C 122703586 IC50 = 10 nM T99340 CYIP81 122703588 IC50 = 10 nM T99340 C5LYJ9 122703599 IC50 = 126 nM T99340 CL7MB6 122703611 IC50 = 16 nM T99340 CJ3RT5 122703613 IC50 = 1.6 nM T99340 C6NT4C 122703637 IC50 = 10 nM T99340 C2TE3N 122703644 IC50 = 9 nM T99340 CP31IH 122703646 IC50 = 200 nM T99340 CIA2M8 122703656 IC50 = 6.3 nM T99340 CX7BC0 122703665 IC50 = 4 nM T99340 CKY5L7 122703666 IC50 = 316 nM T99340 C6R7MN 122703671 IC50 = 10 nM T99340 CAEG59 122703680 IC50 = 10 nM T99340 C8ODW1 122703682 IC50 = 10 nM T99340 CXA83K 122703688 IC50 > 10000 nM T99340 CR1C5H 122703691 IC50 = 4.8 nM T99340 CU7TI5 122703692 IC50 = 10 nM T99340 C27BKA 122703700 IC50 = 1.6 nM T99340 C26JOL 122703705 IC50 = 10 nM T99340 CR75IM 122703716 IC50 = 10 nM T99340 CEG87H 122703723 IC50 = 10 nM T99340 CG7RC6 122703734 IC50 = 398 nM T99340 CK2D8E 122703743 IC50 = 0.5 nM T99340 CZ6R3X 124086061 IC50 = 35 nM T99340 C9XVO7 124086067 IC50 = 10 nM T99340 C7MLB2 124086077 IC50 = 16 nM T99340 CJXY94 124180534 IC50 = 32 nM T99340 CY8JW7 127033346 IC50 > 10000 nM T99340 C3ASY7 127033640 IC50 = 35 nM T99340 C4BKW6 127033641 IC50 = 210 nM T99340 C1KNJ3 127033642 IC50 = 0.2 nM T99340 C1U6TC 130299179 IC50 = 631 nM T99340 C6IZ3V 130299401 IC50 = 3162 nM T99340 CNI1W2 132016672 IC50 = 79 nM T99340 CPF5E3 132471860 Ki = 0.912 nM T99340 CK4HX5 134521326 IC50 = 10 nM T99340 CRT5O7 134521520 IC50 = 8.5 nM T99340 C2E7AT 134521814 IC50 = 1 nM T99340 CG9R3J 134522007 IC50 = 10 nM T99340 CZB75S 134522265 IC50 = 2.5 nM T99340 CSCT10 134536604 IC50 = 7.9 nM T99340 CSL60X 135308861 Ki = 0.912 nM T99340 C0ZQP5 135308877 Ki = 1.738 nM T99340 CS1DF9 135308888 Ki = 13.8 nM T99340 CFX4W3 135308904 Ki = 251.19 nM T99340 CNF6O4 135308906 Ki = 1.778 nM T99340 C6M9FG 135308913 Ki = 2.57 nM T99340 CF1LY8 135308922 Ki = 6918.31 nM T99340 C3XG8C 135308924 Ki = 2.512 nM T99340 C8Z7AU 135308925 Ki = 1.148 nM T99340 C6EW1J 135308927 Ki = 3.467 nM T99340 C8NC5R 135308928 Ki = 2.951 nM T99340 C2C5TL 135308931 Ki = 4265.8 nM T99340 CZP1T3 135308934 Ki = 5.129 nM T99340 CNI5C3 135308946 Ki = 38.02 nM T99340 C8AVZ0 135308996 Ki = 3.89 nM T99340 CSOZ57 135309005 Ki = 7.943 nM T99340 CGFM04 135309027 Ki = 117.49 nM T99340 CQIU03 135309039 Ki = 107.15 nM T99340 CRJ8H5 135309049 Ki = 54.95 nM T99340 C5GAV8 135309066 Ki = 0.8511 nM T99340 CZ53KU 135309069 Ki = 33.88 nM T99340 CA28GI 135309090 Ki = 0.4074 nM T99340 CI8Z2F 135309102 Ki = 1.148 nM T99340 C5E6UB 135314480 IC50 = 39.81 nM T99340 CXC69T 137321158 IC50 = 11 nM T99340 CVGN14 137632484 IC50 = 0.05 nM T99340 C8PV3G 137632977 IC50 > 10000 nM T99340 COL6Q7 137634539 IC50 = 12600 nM T99340 C1FTS9 137634957 IC50 > 10000 nM T99340 C5KYE7 137635049 IC50 = 100 nM T99340 C3EIS6 137635629 IC50 = 0.4 nM T99340 CA8GF2 137637401 IC50 = 2468 nM T99340 CQ32NB 137638108 EC50 > 10000 nM T99340 C58MXE 137640092 IC50 = 2 nM T99340 C5B9NR 137640099 IC50 = 501 nM T99340 CZS13Q 137640111 IC50 = 295 nM T99340 C62DVJ 137640435 EC50 > 3000 nM T99340 CGC9T1 137641614 IC50 > 10000 nM T99340 CESF45 137644276 IC50 = 167 nM T99340 C4TBJ8 137647324 IC50 > 10000 nM T99340 CLP5H9 137647405 IC50 = 0.63 nM T99340 C4JH8A 137647835 IC50 > 10000 nM T99340 CYP70I 137651336 IC50 > 10000 nM T99340 CCK03W 137652965 IC50 > 10000 nM T99340 CKX2D8 137654471 IC50 > 10000 nM T99340 CRH18Z 137656846 IC50 = 178 nM T99340 CP51KG 137657894 IC50 = 1259 nM T99340 CFH52E 137659234 IC50 = 251 nM T99340 C3BCN1 138377545 IC50 = 0.3 nM T99340 CGX92C 138393291 IC50 = 5500 nM T99340 CCT23N 141340950 IC50 > 15000 nM T99340 CTS9Q8 142416001 IC50 = 2.512 nM T99340 CFGH25 142416011 IC50 = 10 nM T99340 C2X1CR 145978863 IC50 = 190 nM T99340 C85UBM 145978937 IC50 = 10 nM T99340 CAW7B1 145980780 IC50 = 468 nM T99340 C43ZUJ 145981140 IC50 = 49 nM T99340 C10HDT 145981335 IC50 = 134 nM T99340 C8DKN3 145981423 IC50 = 94 nM T99340 C89BNR 145982306 IC50 = 531 nM T99340 CO57FT 145982439 IC50 = 3457 nM T99340 CUZQ37 145985171 IC50 = 704 nM T99340 C41ZBR 145986358 IC50 = 105 nM T99340 C4D8HB 145986929 IC50 = 18 nM T99340 C3FN9P 145987011 IC50 = 424 nM T99340 CST1O6 145987202 IC50 = 31 nM T99340 CGM18W 145987557 IC50 = 10 nM T99340 CAC0M7 145988480 IC50 = 13 nM T99340 C7DWU4 145988653 IC50 = 26 nM T99340 CUJL09 145988701 IC50 = 77 nM T99340 C58ULD 145988885 IC50 = 49 nM T99340 CVH28K 145989341 IC50 = 128 nM T99340 COTX64 145989416 IC50 = 2994 nM T99340 C8VND5 145989851 IC50 = 10 nM T99340 C4P8HQ 145990145 IC50 = 264 nM T99340 CZ0RI5 145990208 IC50 = 107 nM T99340 CGF6E4 145990858 IC50 = 17 nM T99340 C96XWF 145991904 IC50 = 28 nM T99340 C3D6OB 145992043 IC50 = 79 nM T99340 CAOQ30 145992060 IC50 = 392 nM T99340 C1NYL4 145993423 IC50 = 634 nM T99340 C05WAM 146344085 IC50 = 90 nM T99340 CN7MS2 154023591 IC50 = 5 nM T99340 CKW68P 155393270 IC50 = 7940 nM T99340 CS0T6E 155510707 IC50 = 17000 nM T99340 C37FPZ 155510738 IC50 > 15000 nM T99340 CX0T1C 155512182 IC50 = 10 nM T99340 C0AUE4 155512296 IC50 = 10 nM T99340 COA84W 155512492 IC50 = 200 nM T99340 C23DJP 155512860 IC50 = 19.95 nM T99340 C2MD1Q 155513187 IC50 > 10000 nM T99340 CZ7K6H 155513660 IC50 > 15000 nM T99340 CC3T0M 155518699 IC50 = 10 nM T99340 CWZ5J8 155519113 IC50 = 5012 nM T99340 CXD9M4 155520427 IC50 = 10 nM T99340 C4FW0B 155522577 IC50 = 6.3 nM T99340 CLW39S 155522794 IC50 = 10 nM T99340 CQIR50 155523679 IC50 = 200 nM T99340 C9M2ZT 155523831 IC50 = 10 nM T99340 CPK67I 155524868 IC50 = 180 nM T99340 CJ3M5T 155524881 IC50 > 1000 nM T99340 CU9H3G 155525351 Ki = 21 nM T99340 C1ICR3 155529856 IC50 > 10000 nM T99340 CIP84Q 155530191 IC50 = 90 nM T99340 C0V9QN 155532882 IC50 > 15000 nM T99340 CTJ84E 155533767 IC50 = 1.3 nM T99340 CQOE59 155534156 IC50 = 310 nM T99340 CF09IN 155535999 IC50 = 10 nM T99340 C8JR2S 155537020 IC50 = 20.8 nM T99340 CSU48D 155537554 IC50 = 10 nM T99340 CZR0J9 155537757 IC50 = 11000 nM T99340 CTP72E 155538424 IC50 = 200 nM T99340 CZ80HO 155547269 IC50 = 10 nM T99340 CSQ28H 155548887 IC50 = 2.5 nM T99340 C5L7HY 155551127 IC50 > 15000 nM T99340 CQ92XF 155552769 IC50 = 126 nM T99340 CDT06B 155555771 IC50 = 600 nM T99340 CL2CH8 155556595 IC50 = 10 nM T99340 C4Z8UW 155569299 IC50 = 1.3 nM T99340 D0K8YD 76332060 IC50 = 16 nM T99340 D0N4LR 53469448 IC50 = 18 nM T28692 D0T9TJ 3034010 IC50 = 66 nM T28692 CBS6H4 2734352 IC50 = 9000 nM T28692 C57UNE 4100861 IC50 = 8000 nM T28692 CP06OA 4197991 IC50 = 9000 nM T28692 C69IFT 4589191 IC50 = 3800 nM T28692 CEB78U 9795865 IC50 = 7000 nM T28692 CG6W8R 9839754 IC50 > 10000 nM T28692 CH0R1M 10038557 IC50 > 50000 nM T28692 CEKX28 10094001 IC50 > 50000 nM T28692 CI70JE 10109540 IC50 = 200 nM T28692 CU21VN 10476544 IC50 > 50000 nM T28692 C0BA2K 11989651 IC50 = 4400 nM T28692 C6D5JN 18172813 IC50 = 1500 nM T28692 CZ7H1I 18525723 IC50 = 9600 nM T28692 C93ZJI 46739726 IC50 = 15000 nM T28692 C1ND3M 54704622 IC50 > 37000 nM T28692 CQ76TF 57391265 IC50 = 15000 nM T28692 C7K6JT 57391611 IC50 = 15000 nM T28692 CA4F1U 57394765 IC50 = 85000 nM T28692 CP03HF 57394766 IC50 = 19000 nM T28692 CTC2Q5 57396517 IC50 > 50000 nM T28692 CR8E0J 57396518 IC50 = 21000 nM T28692 C8P7XU 57396519 IC50 = 55000 nM T28692 C4XS7C 57398310 IC50 = 15000 nM T28692 CTAG79 57399970 IC50 = 25000 nM T28692 CW5DX2 57399971 IC50 = 36000 nM T28692 C1X8DV 57401757 IC50 > 500000 nM T28692 CL3O8E 57401758 IC50 = 120000 nM T28692 C3WCR8 57403489 IC50 = 45000 nM T28692 C3PJ4N 62709758 IC50 > 10000 nM T28692 CZI90M 71744953 IC50 = 1690 nM T28692 CRH31E 72735960 IC50 > 100000 nM T28692 C9GPA3 72735961 IC50 > 33000 nM T28692 C3CT9N 72735962 IC50 = 2560 nM T28692 CPED61 72736167 IC50 > 20000 nM T28692 C0DCX2 72736168 IC50 = 31590 nM T28692 C59NRU 72736169 IC50 > 33000 nM T28692 CH1M8V 72736170 IC50 = 49900 nM T28692 CS7L8X 72736171 IC50 > 33000 nM T28692 CYQ56E 72736172 IC50 > 100000 nM T28692 CA5IR2 72736173 IC50 = 20000 nM T28692 CA3CX9 72736345 IC50 = 76300 nM T28692 C29JMD 72736346 IC50 = 77200 nM T28692 C8WK3T 72736347 IC50 = 45200 nM T28692 C6E9WO 72736348 IC50 > 33000 nM T28692 C52PVL 72736350 IC50 > 100000 nM T28692 CF4HQ3 72736351 IC50 > 100000 nM T28692 CH4GO3 89922162 IC50 = 12000 nM T28692 C3AF7K 90342616 IC50 > 90000 nM T28692 D0F1UD 4589192 IC50 = 1400 nM T28692 D0L8ZG 79799 IC50 = 9000 nM T11451 D0OJ4L 3652 IC50 = 110 nM T11451 CNKJ47 11189680 IC50 = 20 nM T11451 CSZ9E8 11474810 IC50 = 2400 nM T11451 C29BUS 25105690 IC50 = 4.6 nM T11451 CRH90Q 44589003 IC50 = 5200 nM T11451 CJ53QX 44589026 IC50 = 30 nM T11451 CQAJ97 45102599 IC50 = 15 nM T11451 C9ZX1U 45137909 IC50 = 98 nM T11451 CS2C1K 54760105 IC50 = 3.9 nM T11451 CMY13U 54760109 IC50 = 8.6 nM T11451 CC20ZM 54760285 IC50 = 73 nM T11451 CC02GF 54760475 IC50 = 20 nM T11451 CRK2L3 54760476 IC50 = 3.5 nM T11451 CO3MX1 54760671 IC50 = 28 nM T11451 C9CY4L 54760856 IC50 = 13 nM T11451 CRLQ30 54761040 IC50 = 11 nM T11451 CDN2B1 54761215 IC50 = 11 nM T11451 C1C0IR 54761217 IC50 = 16 nM T11451 CQIU13 68246126 IC50 = 35 nM T11451 C1Q6EJ 68341156 IC50 = 27 nM T11451 CO7U3A 68341350 IC50 = 190 nM T11451 CH29GF 71258526 IC50 > 10000 nM T11451 CUC96E 117093964 IC50 = 120 nM T11451 C14VIC 117906466 IC50 = 120 nM T11451 CE0KL1 117906931 IC50 = 73 nM T11451 CR6UL3 117906934 IC50 = 56 nM T11451 C9VN3S 117906987 IC50 = 56 nM T11451 CGT95F 118721661 IC50 = 190 nM T11451 CLK82Y 118721662 IC50 = 84 nM T11451 C08QKE 118721945 IC50 > 1000 nM T11451 C6NTM8 130454358 IC50 = 130 nM T11451 C59JSA 130454361 IC50 = 50 nM T11451 C5DKT7 130454370 IC50 = 28000 nM T11451 C26WUT 130454401 IC50 = 500 nM T11451 C6FHY8 130454431 IC50 = 30 nM T11451 C6B9XI 130454445 IC50 = 18000 nM T11451 CIU01F 130454450 IC50 = 20 nM T11451 CHAE81 130454459 IC50 = 9400 nM T11451 CVEF58 130454467 IC50 = 10000 nM T11451 CG08CU 130454481 IC50 = 20 nM T11451 CTOG04 130454512 IC50 = 50 nM T11451 CY4JT1 130454516 IC50 = 80 nM T11451 CBE8V0 130454542 IC50 = 17000 nM T11451 C8RUV4 130454546 IC50 = 30 nM T11451 C7JNE6 130454574 IC50 = 40 nM T11451 CF06GU 130454579 IC50 = 4800 nM T11451 CBM73C 130454634 IC50 = 20 nM T11451 CXNZ71 130454680 IC50 = 240 nM T11451 CE86DQ 130454681 IC50 = 100 nM T11451 C0U4FJ 130472372 IC50 = 5500 nM T11451 CI84KG 130472422 IC50 = 40 nM T11451 C93TUC 130472439 IC50 = 20 nM T11451 C28LWH 130472440 IC50 = 30 nM T11451 C45BQH 132585194 EC50 = 5660 nM T11451 C14IYS 135545160 IC50 > 50000 nM T11451 CSJ29E 137222695 IC50 = 51000 nM T11451 C1DQ9N 137632868 IC50 = 133 nM T11451 C85BEX 137634734 IC50 = 2100 nM T11451 CD92WT 137635490 IC50 = 21000 nM T11451 C6UK4P 137640101 IC50 = 60 nM T11451 C5UP7W 137640859 IC50 = 99 nM T11451 C1UW7B 137641086 IC50 = 7000 nM T11451 C3GU9A 137642761 IC50 = 830 nM T11451 CN4T8D 137644178 IC50 = 308 nM T11451 CUIL14 137645168 IC50 = 590 nM T11451 CQ0A7B 137647183 IC50 < 50 nM T11451 C8PZN3 137647878 IC50 = 1100 nM T11451 C8LP5F 137653682 IC50 = 2560 nM T11451 C6CDH0 137659544 IC50 = 5100 nM T11451 CXZL91 137661216 IC50 < 50 nM T11451 CSUN37 137661892 IC50 = 100 nM T11451 CWZ59N 145978968 IC50 = 30 nM T11451 CJZ49S 145979394 IC50 = 10200 nM T11451 CGVS82 145986851 IC50 = 200 nM T11451 C6TV1L 145988217 IC50 = 4000 nM T11451 CZ2HG1 145989953 IC50 = 260 nM T11451 C6BMI0 145990319 IC50 = 110 nM T11451 CDQP96 145992257 IC50 = 30 nM T11451 CUG68V 145992733 IC50 = 5000 nM T79068 D00CSQ 5564 Ki = 200 nM T79068 D03KOZ 1549120 IC50 > 200000 nM T79068 D09XQF 3767 IC50 = 8290 nM T79068 D0G3DL 135398735 IC50 = 30 nM T79068 CH7SI8 116119 IC50 = 31500 nM T79068 CY5LO1 258240 IC50 = 38860 nM T79068 CB3J4Y 534602 IC50 = 970 nM T79068 C3B7YT 534606 IC50 = 56500 nM T79068 CZ35WM 542712 IC50 = 4680 nM T79068 CL83PB 571477 IC50 = 3940 nM T79068 C2Z5YG 597131 IC50 = 14500 nM T79068 C2GJ8I 623482 IC50 = 390 nM T79068 C8OU2N 675923 IC50 = 2140 nM T79068 CS2O4Z 675989 IC50 = 3470 nM T79068 C3Z7TS 679013 IC50 = 17620 nM T79068 CF2KO7 681767 IC50 = 9740 nM T79068 CY2G1J 684175 IC50 = 6170 nM T79068 C8DA9R 691843 IC50 = 11480 nM T79068 C1ALD3 702106 IC50 = 7240 nM T79068 CO28PN 702506 IC50 = 6730 nM T79068 C29YIX 708358 IC50 = 3310 nM T79068 CS54OB 711243 IC50 = 52480 nM T79068 C5XDU1 711244 IC50 = 4070 nM T79068 C0PI2W 711536 IC50 = 5010 nM T79068 C7L9IY 717263 IC50 = 10470 nM T79068 C3F9ZU 717273 IC50 = 10000 nM T79068 CB02FT 719451 IC50 > 1000000 nM T79068 C5BX7D 739897 IC50 = 13870 nM T79068 C4ZD8Y 749123 IC50 = 3070 nM T79068 C7PVA3 788974 IC50 = 990 nM T79068 CMG5F0 807901 IC50 = 6260 nM T79068 CWXU43 891794 IC50 > 25000 nM T79068 C9AKN3 892452 IC50 > 25000 nM T79068 CE7NG2 896270 IC50 = 1820 nM T79068 C4XNF7 898412 IC50 > 100000 nM T79068 CRZF52 975517 IC50 = 22120 nM T79068 CW59SG 1012371 IC50 = 1850 nM T79068 CRX97I 1068855 IC50 > 50000 nM T79068 C1UC8W 1070143 IC50 = 6050 nM T79068 CV93DM 1075122 IC50 > 50000 nM T79068 C4SPT9 1108334 IC50 > 100000 nM T79068 CUN24A 1154171 IC50 > 50000 nM T79068 CTDS01 1240234 IC50 = 16030 nM T79068 C37CZY 1240238 IC50 > 50000 nM T79068 CAVG24 1292455 IC50 > 100000 nM T79068 CS15YR 1393330 IC50 = 7830 nM T79068 C4AS2B 1988345 IC50 > 100000 nM T79068 CMB4W3 2184078 IC50 = 19960 nM T79068 CO6PH8 2236231 IC50 = 10720 nM T79068 CO7V3K 2275922 IC50 > 50000 nM T79068 C4OAJ2 2838469 IC50 = 15470 nM T79068 CC7F6V 2844150 IC50 = 10050 nM T79068 CEYC67 2855970 IC50 = 73580 nM T79068 C53IHK 2856144 IC50 > 100000 nM T79068 CM5XV4 2856288 IC50 = 34880 nM T79068 CEX92I 2872768 IC50 > 100000 nM T79068 C1WZ5P 2883369 IC50 = 10590 nM T79068 C38UNC 2883437 IC50 = 28020 nM T79068 C52KDN 2883505 IC50 = 10660 nM T79068 C4RA1M 2883636 IC50 > 100000 nM T79068 C4ZSY9 2883637 IC50 > 100000 nM T79068 CU23DP 2883815 IC50 > 100000 nM T79068 CEKV85 2890189 IC50 > 100000 nM T79068 C49OTS 2902416 IC50 = 13550 nM T79068 C3VBO2 2926591 IC50 > 100000 nM T79068 CP0JS5 2926817 IC50 > 100000 nM T79068 C5LI7X 2927358 IC50 = 56020 nM T79068 CB05RK 2942596 IC50 > 100000 nM T79068 C2FAS9 2947371 IC50 > 100000 nM T79068 CB38MC 2947665 IC50 > 100000 nM T79068 COIC68 2948561 IC50 = 29230 nM T79068 CEAL91 2966678 IC50 = 31370 nM T79068 CTNL82 2984958 IC50 > 75000 nM T79068 CHRS80 2985043 IC50 > 100000 nM T79068 C4UBW9 2986000 IC50 = 23120 nM T79068 CDW6Z1 2986297 IC50 = 14830 nM T79068 CQ6A9O 2986544 IC50 = 1600 nM T79068 C85CBZ 2986800 IC50 > 100000 nM T79068 C5S3CL 2989189 IC50 = 5100 nM T79068 CP64DV 2989420 IC50 > 100000 nM T79068 C45MRK 2991467 IC50 = 16790 nM T79068 CH37UN 3037036 Ki = 4800 nM T79068 CL2A6G 3105210 IC50 > 100000 nM T79068 CA40TK 3112066 IC50 = 1350 nM T79068 CZP40A 3112067 IC50 = 890 nM T79068 C2WU8M 3149415 IC50 > 100000 nM T79068 CDX79Z 3161308 IC50 = 1490 nM T79068 C3P1BI 3412846 IC50 = 2900 nM T79068 CR0VI2 3412850 IC50 = 397 nM T79068 CK1FO0 3941420 IC50 = 37410 nM T79068 C8XEM4 4006554 IC50 = 9430 nM T79068 CHCT27 8366407 IC50 = 90 nM T79068 CUZ1E6 9003925 IC50 = 222 nM T79068 C1S3HK 9003927 IC50 = 1690 nM T79068 CL2F6U 9378917 IC50 = 2040 nM T79068 C3MFP1 9517691 IC50 = 361 nM T79068 CD74UH 10249327 IC50 = 75000 nM T79068 CAU7G8 16072548 IC50 = 270 nM T79068 CT8FG9 16072549 IC50 = 140 nM T79068 CU75NH 16072550 IC50 = 620 nM T79068 CQK16R 16072551 IC50 = 850 nM T79068 CX6ZJ9 16072552 IC50 = 320 nM T79068 C4FUP7 16072553 IC50 = 750 nM T79068 CSE69C 16072554 IC50 = 2570 nM T79068 C6Z9NJ 16072555 IC50 = 3390 nM T79068 C5YJ0B 16072556 IC50 = 410 nM T79068 CB2U7Z 16072557 IC50 = 390 nM T79068 C2NFI6 16077255 IC50 = 3510 nM T79068 CA69KZ 16077257 IC50 = 3140 nM T79068 C1FZ7N 16077258 IC50 = 1300 nM T79068 C3ER5H 16077259 IC50 = 3670 nM T79068 C1XDF3 16077262 IC50 = 4470 nM T79068 CG81MN 16077263 IC50 = 5180 nM T79068 CM2GS7 16077264 IC50 = 6410 nM T79068 CY4IC8 16077266 IC50 = 5510 nM T79068 CR9TI7 16077274 IC50 = 1290 nM T79068 CL1W5K 16090567 IC50 = 1390 nM T79068 CRP17Q 16727110 IC50 = 22 nM T79068 C2ASO7 17005290 IC50 = 1000 nM T79068 CZ0K2N 17312855 IC50 = 1890 nM T79068 C28UOD 17549537 IC50 = 7620 nM T79068 C05GLR 17683363 IC50 > 50000 nM T79068 C20YLR 22600366 Ki = 2100 nM T79068 CUY5O6 23647179 IC50 = 460 nM T79068 C9Q1GW 23647180 IC50 = 850 nM T79068 CF2BW9 25093354 IC50 = 1040 nM T79068 C0UR1F 44417313 IC50 = 5550 nM T79068 C1OBT4 44441987 IC50 = 27000 nM T79068 C6S9MB 44450005 Ki = 1 nM T79068 CUX48V 44450006 Ki = 1 nM T79068 CD0K8I 44450030 Ki = 1 nM T79068 CTB6O7 44450031 Ki = 1 nM T79068 C93HZW 44450032 Ki = 1 nM T79068 CF45GX 44450056 Ki = 1 nM T79068 CIRP08 44450057 Ki = 1 nM T79068 C4OCA3 44450058 Ki = 1 nM T79068 CZ2UD7 45265853 IC50 = 62 nM T79068 CO9W4T 45268587 IC50 = 5130 nM T79068 C7QN5Z 45272005 IC50 = 5010 nM T79068 C9J6ZI 45272827 IC50 = 10960 nM T79068 C1TQV7 46927949 IC50 = 3 nM T79068 CZSH81 46946547 IC50 = 4 nM T79068 C5QYL7 55363227 IC50 > 50000 nM T79068 CGI05U 71624761 Ki = 71000 nM T79068 CEAO21 71717931 Ki = 0.75 nM T79068 C0KMW2 72713535 IC50 = 234 nM T79068 CLZ82F 72713536 IC50 = 30 nM T79068 CJA8Q5 72713752 IC50 = 200 nM T79068 C1FV3N 72713753 IC50 < 2 nM T79068 C7JKX5 72713754 IC50 < 2 nM T79068 C6T8FE 72713755 IC50 = 970 nM T79068 CK4N6B 72713756 IC50 = 400 nM T79068 CVA1J0 72713757 IC50 = 34000 nM T79068 C8QEJ3 72725792 IC50 = 34 nM T79068 CF8WR0 76310895 IC50 > 1000 nM T79068 CWJQ73 76314523 IC50 = 40 nM T79068 CSJ71E 76314524 IC50 = 26 nM T79068 CX60CH 76314525 IC50 > 1000 nM T79068 CQ0HM6 76314526 IC50 = 4 nM T79068 CJ8GL6 76314527 IC50 = 5 nM T79068 CGR21C 76314528 IC50 = 22 nM T79068 CKZT86 76314529 IC50 = 11 nM T79068 CQFG10 76314530 IC50 = 4 nM T79068 CQ6YT8 76314531 IC50 = 74 nM T79068 C5AD8G 76314532 IC50 = 121 nM T79068 C9B7JI 76314533 IC50 = 215 nM T79068 C8C5MV 76318088 IC50 = 2 nM T79068 C3OE1K 76318089 IC50 = 3 nM T79068 C4F8NK 76318104 IC50 = 112 nM T79068 CF4U8J 76318105 IC50 = 25 nM T79068 CA3KW2 76318106 IC50 = 3 nM T79068 CQ9D8P 76318107 IC50 = 5 nM T79068 CUX6N5 76318108 IC50 = 32 nM T79068 C84VFR 76318109 IC50 > 1000 nM T79068 CJ9F8Q 76318110 IC50 = 46 nM T79068 CJVF30 76318111 IC50 = 21 nM T79068 C1GB2V 76318112 IC50 = 14 nM T79068 CARF53 76321796 IC50 = 45 nM T79068 CPG4V9 76321797 IC50 = 17 nM T79068 CWF5T2 76321798 IC50 = 15 nM T79068 C79AGH 76321799 IC50 = 120 nM T79068 CCNZ57 76321800 IC50 = 948 nM T79068 C5PU3Z 76321801 IC50 = 170 nM T79068 C4XY8N 76321802 IC50 = 22 nM T79068 C3HVK8 76321803 IC50 = 20 nM T79068 CI76CV 76325437 IC50 = 11 nM T79068 CIS2G3 76325438 IC50 = 3 nM T79068 C6BWY3 76325439 IC50 > 1000 nM T79068 C6PLI0 76328070 IC50 = 20 nM T79068 CLAH84 76328962 IC50 = 4 nM T79068 C0KG4J 76328976 IC50 = 41 nM T79068 C89CTR 76328977 IC50 = 7 nM T79068 CE7Q6G 76328978 IC50 = 3 nM T79068 CW7RL1 76328979 IC50 = 12 nM T79068 CEF34Y 76332639 IC50 = 4 nM T79068 CS8Z6N 76332645 IC50 = 2 nM T79068 CN7DK9 76332646 IC50 = 80 nM T79068 CBF76O 76332647 IC50 = 5 nM T79068 CYL50Z 76332648 IC50 = 22 nM T79068 CM80JY 76332649 IC50 = 35 nM T79068 C2I6YG 76332650 IC50 = 18 nM T79068 C1NP4B 76332651 IC50 = 7 nM T79068 CRZ3U0 76332652 IC50 = 1290 nM T79068 C1IQW7 76332653 IC50 = 440 nM T79068 CVBO81 76336253 IC50 = 42 nM T79068 C9B2EA 76336254 IC50 = 9 nM T79068 CMO2W7 76336255 IC50 = 6 nM T79068 CF2SR1 76336256 IC50 = 9 nM T79068 CM8PO0 76336257 IC50 = 21 nM T79068 C9D5NX 76336258 IC50 = 5 nM T79068 C5MWL1 101879982 IC50 = 5120 nM T79068 C4DK5L 118709527 IC50 > 50000 nM T79068 CP65YN 118713598 IC50 = 3120 nM T79068 C0FPC3 118714489 IC50 > 100000 nM T79068 CMDG59 118714492 IC50 > 100000 nM T79068 CZ0F1B 118717393 IC50 = 8230 nM T79068 CT72VB 118717395 IC50 = 6820 nM T79068 CL0HY3 118717396 IC50 = 8900 nM T79068 CXE4D9 118725819 IC50 > 50000 nM T79068 CV0ON9 118725820 IC50 = 250 nM T79068 CI2T9Y 118725821 IC50 = 5990 nM T79068 CGE72I 118725822 IC50 = 240 nM T79068 CQW18I 118725823 IC50 = 1570 nM T79068 CL9PS1 118725824 IC50 = 9770 nM T79068 C4A0RN 118725825 IC50 > 50000 nM T79068 CD83NI 118725826 IC50 > 50000 nM T79068 CGLY68 118725827 IC50 > 50000 nM T79068 CS51EW 135658044 IC50 = 17780 nM T79068 C7K3JS 146020572 IC50 = 310 nM T79068 CV2O5J 155514214 IC50 = 6000 nM T79068 CTD72C 155517063 IC50 = 4000 nM T79068 CKY1T8 155517820 IC50 = 2820 nM T79068 C21KID 155536460 IC50 = 9000 nM T79068 CQ56AI 155538508 IC50 = 11600 nM T79068 CKS05E 155540873 IC50 = 16800 nM T79068 C5S1BT 155542700 IC50 = 28100 nM T79068 CN67SO 155550889 IC50 = 22600 nM T79068 COTS64 155551046 IC50 = 55000 nM T79068 CP9W0R 155551049 IC50 = 22000 nM T79068 CR9OG4 155551781 IC50 = 50100 nM T79068 C1KXF4 155552900 IC50 = 40200 nM T79068 CVO8R1 155554323 IC50 = 43500 nM T79068 C9RU6S 155554664 IC50 = 25800 nM T79068 C35AKQ 155555440 IC50 = 8240 nM T79068 CU1G4Q 155555508 IC50 = 23900 nM T79068 C25RBL 155555688 IC50 = 15300 nM T79068 C57WML 155556087 IC50 = 3120 nM T79068 CE43LT 155557034 IC50 = 12100 nM T79068 C06ETK 155557211 IC50 = 35300 nM T79068 CMG4N0 155559921 IC50 = 47300 nM T79068 CW50RA 155560078 IC50 = 17400 nM T79068 C3T8BX 155560664 IC50 = 20100 nM T79068 CPUS15 155562689 IC50 = 17500 nM T79068 C5SKX6 155563240 IC50 = 7840 nM T79068 CN54ME 155565487 IC50 = 2550 nM T79068 CLCY25 155567123 IC50 = 5020 nM T79068 CY5B2C 155567303 IC50 = 16500 nM T79068 C5AXF8 155568250 IC50 = 250 nM T79068 D01EFQ 44450157 Ki = 1 nM T79068 D01MLQ 667749 IC50 = 14110 nM T79068 D04BHQ 577479 IC50 = 10470 nM T79068 D04XUV 44450123 Ki = 1 nM T79068 D05DRQ 675939 IC50 = 4370 nM T79068 D05MLT 44450091 Ki = 1 nM T79068 D05NWQ 711259 IC50 = 19950 nM T79068 D05OQF 711431 IC50 = 6170 nM T79068 D05SWR 711551 IC50 = 13800 nM T79068 D07UTV 711434 IC50 = 12020 nM T79068 D08AFZ 1415427 IC50 = 5160 nM T79068 D08KWS 5274977 Ki = 1 nM T79068 D08VHO 44450159 Ki = 1 nM T79068 D08ZCM 5274979 Ki = 1 nM T79068 D09JHY 44450061 Ki = 1 nM T79068 D09LQF 45272830 IC50 = 1350 nM T79068 D0E9CT 447767 IC50 = 200 nM T79068 D0FI4X 44450095 Ki = 1 nM T79068 D0G7MC 44450183 Ki = 1 nM T79068 D0I1RG 749125 IC50 = 16640 nM T79068 D0IA7R 44450094 Ki = 1 nM T79068 D0J1PL 44450124 Ki = 1 nM T79068 D0JQ7W 675658 IC50 = 9550 nM T79068 D0K9LT 16063378 Ki = 1 nM T79068 D0K9LV 44450156 Ki = 1 nM T79068 D0M0EE 44450092 Ki = 1 nM T79068 D0M5EU 1378917 IC50 = 7390 nM T79068 D0N0IC 711547 IC50 = 7080 nM T79068 D0N4IT 695266 IC50 = 19950 nM T79068 D0O1BT 44450125 Ki = 1 nM T79068 D0P9AP 44450160 Ki = 1 nM T79068 D0TH7L 44450122 Ki = 1 nM T79068 D0X8JE 44450093 Ki = 1 nM T79068 D0YK5U 711291 IC50 = 8710 nM T79068 D0ZM1Q 814705 IC50 = 7740 nM T41141 D0V3YT 10324367 IC50 = 760 nM T41141 D0X9CH 3010818 IC50 = 3500 nM T41141 D0J6AU 10152654 Ki = 1258.93 nM T41141 D0HM5J 118253852 IC50 > 20000 nM T41141 D01LNG 10201696 IC50 = 48 nM T41141 D04ZIJ 5478883 IC50 = 800 nM T41141 D0T5PH 6918602 Ki = 0.068 nM T41141 CD3P2Z 8857 IC50 > 10000 nM T41141 CU27VZ 12050 IC50 > 100000 nM T41141 C05HLN 26030 Ki = 48000 nM T41141 CIF9A2 95706 IC50 = 6800 nM T41141 CVZP51 125190 IC50 = 50 nM T41141 C5YNV4 161091 IC50 = 2600 nM T41141 CV8A4D 163098 IC50 = 600 nM T41141 C4U5MD 202918 IC50 > 50000 nM T41141 C62DWI 231061 IC50 = 43000 nM T41141 C8OHY9 254021 IC50 = 600 nM T41141 C07JLH 404672 Ki = 8700 nM T41141 CN67CR 555078 IC50 > 100000 nM T41141 CRY54Z 690107 IC50 > 10000 nM T41141 C31BIK 832505 IC50 = 15000 nM T41141 C65UJT 980235 IC50 = 31630 nM T41141 C25SXA 1440071 IC50 = 24390 nM T41141 C9RQ2F 2848907 IC50 = 1600 nM T41141 CT8KV2 3001308 IC50 > 10000 nM T41141 CTE79D 3011892 Ki = 760000 nM T41141 C08KQP 3032999 IC50 > 10000 nM T41141 CWU18B 3082865 Ki = 1.3 nM T41141 CU43OY 3088969 Ki = 134000 nM T41141 C3G8IK 3731185 IC50 = 170 nM T41141 CKM1S9 3827422 IC50 = 510 nM T41141 CMW5A9 4430623 Ki = 245000 nM T41141 C2ZN0V 4479093 IC50 = 90000 nM T41141 CR2ND4 5287468 Ki = 2.2 nM T41141 CW6D7Z 5287498 IC50 = 160000 nM T41141 CB6H0T 5287549 Ki = 0.49 nM T41141 CESY50 5288259 IC50 = 330 nM T41141 C6YF4B 5288616 IC50 = 89 nM T41141 CFM6E4 5288618 IC50 = 82 nM T41141 C9E1UW 5288633 Ki = 700 nM T41141 CN3RY0 5289345 Ki = 340 nM T41141 CWOL57 5339865 IC50 = 45000 nM T41141 CR6B4P 5465605 IC50 > 10000 nM T41141 C3B5YE 5728928 IC50 > 100000 nM T41141 C57VBE 5762376 IC50 > 10000 nM T41141 CW94RA 5897251 IC50 = 98680 nM T41141 C3KI5C 5910205 IC50 > 10000 nM T41141 C1DAZ6 6420159 Ki > 10000 nM T41141 CD51MJ 6442675 IC50 = 30340 nM T41141 CQM64S 6610323 IC50 = 1.9 nM T41141 C0XQP7 6917747 IC50 > 100000 nM T41141 C9BGP6 7020268 Ki = 16000 nM T41141 C7WP6J 8194707 IC50 > 100000 nM T41141 CUXQ12 8832875 IC50 = 29810 nM T41141 C2GV5W 8854795 IC50 > 100000 nM T41141 CN26IL 9547980 Ki > 30000 nM T41141 CF40ZX 9562299 IC50 > 10000 nM T41141 C3QN6S 9571439 IC50 > 10000 nM T41141 CLE53W 9580655 IC50 = 741 nM T41141 CC2ZY8 9580662 IC50 = 228 nM T41141 CT3Y9G 9580665 IC50 = 369 nM T41141 CE42MQ 9809035 Ki = 28.8 nM T41141 CB32AH 9812750 IC50 = 430 nM T41141 C4UE3W 9813935 IC50 = 11500 nM T41141 CQ1NG7 9815041 IC50 = 498 nM T41141 CIX3A6 9816412 IC50 = 80 nM T41141 COBW38 9821383 IC50 = 3090 nM T41141 C9F7PL 9825191 Ki = 22300 nM T41141 C0N4DH 9825355 IC50 = 1800 nM T41141 CN51PR 9829299 Ki = 1000 nM T41141 CK7B2P 9829646 IC50 = 20 nM T41141 C2AI0Z 9834360 IC50 = 1750 nM T41141 CNU47F 9834637 IC50 = 20000 nM T41141 CLND75 9835685 IC50 = 850 nM T41141 CLQ92U 9848147 IC50 = 10000 nM T41141 C8TL5X 9855884 IC50 = 650 nM T41141 CVS7N2 9877581 IC50 = 100 nM T41141 CC3X2P 9877623 IC50 = 100 nM T41141 CO0PD1 9883178 IC50 = 300 nM T41141 CCAI25 9886751 IC50 = 15 nM T41141 C0NM3D 9887557 IC50 = 990 nM T41141 CGA91J 9890145 IC50 > 10000 nM T41141 C8P5LN 9891030 Ki = 190 nM T41141 C8HI1R 9891108 IC50 = 1400 nM T41141 C5L4YE 9893225 IC50 = 1.2 nM T41141 COK50T 9895628 IC50 = 18 nM T41141 CIBS75 9899272 IC50 = 150 nM T41141 C2JCM5 9902742 IC50 = 400 nM T41141 C5XS2F 9904539 Ki = 700 nM T41141 CALH63 9908450 IC50 = 320 nM T41141 C7WKG9 9913437 IC50 > 10000 nM T41141 C78CYD 9920989 IC50 = 23000 nM T41141 CXD2Y6 9926586 IC50 = 500 nM T41141 CNR6D5 9948720 IC50 = 55 nM T41141 C0PJ2U 9964915 IC50 = 50 nM T41141 C4WFJ2 9980678 Ki = 640 nM T41141 CBNR45 9980918 IC50 > 1000 nM T41141 CHN80D 9981917 IC50 > 10000 nM T41141 C1F4BA 9984481 IC50 = 10.7 nM T41141 C69FCE 9987052 Ki = 930 nM T41141 C7P6JO 10004326 IC50 > 1000 nM T41141 C40APB 10005577 IC50 > 1000 nM T41141 CI96RJ 10008050 IC50 = 48.7 nM T41141 CXY9N8 10024008 IC50 > 1000 nM T41141 CLB5G0 10025017 IC50 = 410 nM T41141 C4NW7I 10026902 IC50 > 1000 nM T41141 C0SJY5 10031327 IC50 = 139 nM T41141 C68HGW 10047261 IC50 = 352 nM T41141 C8F7MU 10047536 IC50 > 1000 nM T41141 C2N9CS 10062713 IC50 = 12 nM T41141 C1QB5U 10063343 IC50 = 2900 nM T41141 C5KR4U 10068161 IC50 = 4300 nM T41141 C1IZ3A 10075688 Ki = 0.6 nM T41141 CV29YC 10076076 IC50 = 1700 nM T41141 CHA42Q 10097070 IC50 > 10000 nM T41141 CD6L1T 10098422 Ki = 19 nM T41141 C8FPB5 10098917 IC50 = 1 nM T41141 CSO9B2 10099774 Ki = 120 nM T41141 CA5N3E 10111943 IC50 = 115 nM T41141 C57JDN 10118049 IC50 = 11.5 nM T41141 CFC3Q8 10120133 IC50 = 33000 nM T41141 C6AZ3B 10120903 IC50 = 1000000 nM T41141 C97NJR 10121949 Ki = 11000 nM T41141 C7XOA0 10127183 IC50 = 344 nM T41141 CSO96K 10127748 IC50 = 1300 nM T41141 CKZ15P 10129236 IC50 = 680 nM T41141 CJ79ZX 10138553 IC50 = 1667 nM T41141 CY6PU1 10143615 Ki = 3.9 nM T41141 CLID02 10144235 Ki = 19000 nM T41141 CQ3YD8 10150891 IC50 = 1475 nM T41141 C8DQG0 10154619 IC50 > 10000 nM T41141 C9VFI4 10161284 IC50 = 24000 nM T41141 C1Q2EX 10164497 Ki = 300 nM T41141 CDX7R4 10164961 IC50 = 17000 nM T41141 C5B1HM 10165557 IC50 = 10000 nM T41141 C09ALX 10165785 Ki = 0.04 nM T41141 CR62PT 10165786 Ki = 52 nM T41141 CTJ7R3 10166544 IC50 = 36000 nM T41141 CDRE91 10167323 Ki = 37000 nM T41141 CZ1A8U 10173731 IC50 = 524 nM T41141 C5NEX6 10174161 IC50 = 2200 nM T41141 C1YR4T 10174359 IC50 = 1300 nM T41141 CD4G7F 10179450 IC50 = 108 nM T41141 CTON03 10179451 IC50 = 2101 nM T41141 C07GUT 10184761 Ki = 390 nM T41141 C4M3SG 10186046 IC50 = 3800000 nM T41141 CCO7A6 10187105 Ki = 10000 nM T41141 CP2M1T 10187189 Ki = 4.2 nM T41141 C9WTI5 10187190 Ki = 45 nM T41141 C0SF7U 10187920 IC50 = 10000 nM T41141 CKZ1A0 10194354 IC50 = 80 nM T41141 CZD7A6 10194447 IC50 = 878 nM T41141 CA2UH4 10194634 IC50 = 887 nM T41141 CO7XD6 10198366 IC50 = 6 nM T41141 C5T8PK 10198752 IC50 = 54 nM T41141 CQ8YM3 10199981 Ki = 9600 nM T41141 CL9DW3 10200425 IC50 = 4804 nM T41141 CS3IP7 10210867 IC50 = 190000 nM T41141 C1WL9J 10211340 Ki = 1400 nM T41141 CV0CI4 10216098 Ki = 20 nM T41141 C1F9SP 10216231 IC50 = 1857 nM T41141 C1Y3QZ 10216510 IC50 = 1670 nM T41141 C5GSN6 10216511 IC50 = 2792 nM T41141 CT8K5D 10231379 IC50 = 8700 nM T41141 C4OZ5K 10231447 IC50 = 69000 nM T41141 CJBI61 10237771 IC50 = 13 nM T41141 CFI43Z 10238903 IC50 = 470 nM T41141 CORW86 10247897 IC50 = 150 nM T41141 CEQ21I 10249499 IC50 > 1000 nM T41141 C6A8NV 10252643 Ki = 81 nM T41141 C9SOH2 10271564 IC50 = 1682 nM T41141 CKX0R7 10287617 IC50 = 34 nM T41141 CUW38E 10288162 IC50 = 1001 nM T41141 CX23AL 10288163 IC50 = 3002 nM T41141 CY7DQ2 10288811 IC50 = 1600 nM T41141 CV9LB1 10302710 IC50 = 17000 nM T41141 CUQ2R3 10303526 IC50 = 240000 nM T41141 CV5S7B 10303657 IC50 = 1000000 nM T41141 CZR02J 10303878 Ki = 7500 nM T41141 CPT49O 10310362 IC50 = 3047 nM T41141 CO0GQ8 10313520 IC50 = 450 nM T41141 C9DN6G 10325113 IC50 = 31.9 nM T41141 CXN4D2 10327819 Ki = 70 nM T41141 C59ZDR 10337631 IC50 > 1000 nM T41141 C2GLK6 10346121 IC50 = 0.1 nM T41141 C7D9XB 10363069 IC50 = 22000 nM T41141 CDY26B 10366413 Ki = 6100 nM T41141 CDX2C8 10367993 IC50 > 1000 nM T41141 CYF98Z 10368089 IC50 = 2300 nM T41141 CD9ZI0 10373289 Ki = 720 nM T41141 CX7S8A 10392779 IC50 = 10.8 nM T41141 C7LU1Z 10395274 Ki = 74000 nM T41141 CF7O6A 10409137 IC50 > 20000 nM T41141 C41JUO 10414118 IC50 = 3.8 nM T41141 CDVZ19 10431266 Ki = 6800 nM T41141 CCD1B8 10433014 IC50 = 7 nM T41141 C8DTH3 10436731 IC50 = 554 nM T41141 C57DYJ 10437715 Ki = 2 nM T41141 CN18SE 10456222 Ki = 0.47 nM T41141 C06QJW 10457653 IC50 = 0.1 nM T41141 CK9PX5 10461097 Ki > 1000 nM T41141 C6KJM2 10461790 Ki = 154000 nM T41141 C5M7BL 10471316 IC50 = 1000 nM T41141 CXD68E 10473874 IC50 = 190 nM T41141 C32MAD 10482525 IC50 < 0.4 nM T41141 CW7V0M 10496067 IC50 > 1000 nM T41141 C1MX2S 10499322 Ki = 250 nM T41141 CHTL13 10507714 Ki = 39 nM T41141 CZ80TL 10507960 Ki > 1000 nM T41141 CGA7D1 10515827 IC50 = 350 nM T41141 C25HQJ 10522795 Ki > 1000 nM T41141 C0UBF5 10524384 Ki = 580 nM T41141 CZUA37 10531571 Ki > 1000 nM T41141 COP6I9 10566003 IC50 = 200 nM T41141 CR54HQ 10569603 Ki > 10000 nM T41141 C8U1RQ 10593841 Ki = 2600 nM T41141 CM29WH 10663100 IC50 = 290 nM T41141 CJ7U3O 10668284 IC50 > 10000 nM T41141 CRL23A 10674588 Ki > 1000 nM T41141 C9PY4N 10690022 Ki = 850 nM T41141 CKO6L0 10698950 Ki = 16 nM T41141 CP2WG8 10716501 IC50 = 32 nM T41141 C5E8FN 10793407 Ki = 290 nM T41141 C9AIY1 10793962 Ki = 49 nM T41141 C9XI7T 10804795 IC50 = 900 nM T41141 CQ08YK 10807774 Ki > 1000 nM T41141 CHC3F0 10817683 Ki = 290 nM T41141 CZ4V0F 10832380 Ki > 10000 nM T41141 C78VEK 10837067 Ki > 1000 nM T41141 C1BT8R 10853144 IC50 = 110 nM T41141 CBWJ85 10862359 IC50 = 6273 nM T41141 CNVG58 10875013 IC50 > 10000 nM T41141 CMO9Y1 10886114 Ki = 9.6 nM T41141 C7ZNC2 10892596 IC50 = 170 nM T41141 CZK49P 10893343 IC50 = 2710 nM T41141 CBJ1I7 10902914 IC50 > 10000 nM T41141 CA30HS 10905508 IC50 > 10000 nM T41141 CA9ZC6 10907387 Ki = 44 nM T41141 C5X6NA 10924832 IC50 = 5583 nM T41141 CZG37Y 10938664 IC50 > 10000 nM T41141 CA72YH 10949332 IC50 = 31 nM T41141 CL7W4P 10960628 IC50 = 800 nM T41141 CW1L5K 10960899 IC50 = 1500 nM T41141 CR0P8J 10971179 IC50 > 10000 nM T41141 CK9E8W 10972182 IC50 = 3907 nM T41141 C6ZOI1 10979734 IC50 = 5952 nM T41141 CCFA87 10983274 IC50 = 80 nM T41141 CA3NG9 10993428 IC50 > 10000 nM T41141 C7BI2T 11009218 IC50 = 2600 nM T41141 CM9Z5T 11012257 IC50 = 825 nM T41141 C5XHI0 11014664 IC50 = 1593 nM T41141 C56FMI 11027472 Ki = 7.9 nM T41141 CL19TE 11028356 Ki = 2.8 nM T41141 CY72BF 11034349 IC50 > 10000 nM T41141 CQXP76 11050104 Ki = 144.4 nM T41141 CMP6K1 11071803 Ki = 4.7 nM T41141 CY3V4J 11080121 IC50 = 6 nM T41141 C0PSR8 11081485 IC50 > 10000 nM T41141 C5WY1H 11082075 IC50 < 30 nM T41141 CMC63T 11113842 Ki = 28.8 nM T41141 CQ4L0T 11122768 IC50 = 50 nM T41141 CQK6U4 11144121 IC50 = 4000 nM T41141 CDR7A6 11155973 Ki = 24 nM T41141 C8EAL0 11156785 Ki = 193 nM T41141 C9SN1Q 11157631 Ki = 98 nM T41141 CH41OF 11157632 Ki = 1520 nM T41141 C61AIQ 11168385 Ki = 588 nM T41141 CAI94Q 11168613 Ki = 372 nM T41141 C2VJG7 11178623 Ki = 541 nM T41141 CMDU74 11180007 Ki = 11530 nM T41141 CS90MB 11191512 Ki = 2678 nM T41141 CN0F8E 11199915 IC50 = 1270 nM T41141 C2H4GP 11200735 Ki = 11 nM T41141 CTCX89 11203484 Ki > 65000 nM T41141 C17UIX 11203679 IC50 = 560 nM T41141 C7SOL0 11224927 Ki = 7460 nM T41141 CM8ZV1 11225780 Ki = 18900 nM T41141 CLC2X1 11226457 Ki = 1800 nM T41141 C0JO5R 11238059 Ki > 100000 nM T41141 C3T1LM 11238468 Ki > 50000 nM T41141 C5VY1E 11247716 Ki = 9040 nM T41141 CLA6J3 11249688 Ki > 37000 nM T41141 CRXU26 11250282 Ki = 2310 nM T41141 CHK9N2 11261516 Ki = 3520 nM T41141 C8F2ZN 11269453 IC50 > 1000 nM T41141 CIFQ06 11273375 Ki = 5 nM T41141 C15XUE 11283547 Ki = 11530 nM T41141 CCH6N4 11283555 IC50 = 456 nM T41141 CM86BP 11294094 Ki = 11800 nM T41141 CFU50G 11294227 Ki = 2830 nM T41141 CV86IB 11295906 Ki > 11000 nM T41141 CZX89I 11305296 Ki = 8370 nM T41141 CR2T5B 11305867 Ki = 914 nM T41141 CU6Z0F 11306593 Ki > 37000 nM T41141 CEC0A2 11316876 Ki > 10000 nM T41141 CDYL91 11327594 Ki > 100000 nM T41141 CP5MI6 11329727 Ki > 30000 nM T41141 CD70PA 11341599 Ki = 108 nM T41141 C5X1VW 11351327 IC50 = 62 nM T41141 CFJ70U 11353015 Ki = 4670 nM T41141 C9W0TB 11375856 Ki > 100000 nM T41141 C7NQX3 11375955 Ki = 777 nM T41141 CH4I3T 11375956 IC50 = 230 nM T41141 C34DFQ 11376188 Ki > 70000 nM T41141 CAL7B2 11376611 Ki > 100000 nM T41141 COV1F4 11387157 Ki = 48370 nM T41141 CEW0F3 11387421 Ki = 4080 nM T41141 C3DQL2 11396020 Ki > 30000 nM T41141 C4QM7I 11396148 Ki > 10000 nM T41141 CER2V8 11397519 Ki = 1730 nM T41141 C4ZLU9 11397590 Ki > 30000 nM T41141 C7RFC5 11398171 Ki = 267 nM T41141 CI3HK2 11409407 Ki = 849 nM T41141 CO4Y3H 11410560 Ki > 100000 nM T41141 CU4P8A 11418931 Ki = 17 nM T41141 C56SXA 11419952 Ki = 1150 nM T41141 CGD1K4 11421700 Ki = 17700 nM T41141 CILJ37 11431699 Ki > 30000 nM T41141 CM2VQ6 11431993 Ki = 9670 nM T41141 C19YRB 11432272 Ki = 8990 nM T41141 C72PFO 11432501 Ki = 123 nM T41141 C65ASH 11432773 Ki > 100000 nM T41141 CQRB45 11433280 Ki = 636 nM T41141 CQIP48 11439739 IC50 = 76 nM T41141 CH9ZA7 11443990 Ki = 199 nM T41141 C1AT2Z 11453155 IC50 = 68 nM T41141 CL53MS 11456165 Ki > 100000 nM T41141 CME32S 11456379 Ki > 100000 nM T41141 C0O8MK 11464526 IC50 = 44 nM T41141 C5N3BV 11466327 Ki > 10000 nM T41141 CV43WB 11466677 Ki = 285 nM T41141 CM59AQ 11466845 Ki = 1180 nM T41141 CL1D2Z 11471738 IC50 = 1711 nM T41141 C0ZK5I 11477975 Ki = 150 nM T41141 C9U0YI 11478637 Ki = 3936 nM T41141 CBC8U6 11490230 Ki = 369 nM T41141 CM41QW 11494775 Ki = 54 nM T41141 CT8S4U 11496335 Ki = 900 nM T41141 C5CL9A 11496988 Ki > 15000 nM T41141 CC92RV 11501571 IC50 = 32000 nM T41141 CFI8L5 11502586 IC50 = 150 nM T41141 CK5JM6 11503223 IC50 = 2274 nM T41141 CY4A7V 11504785 Ki = 5 nM T41141 C3Q7BE 11504819 Ki = 150 nM T41141 CCH09G 11507712 Ki > 150000 nM T41141 CHI9N5 11512144 Ki = 8800 nM T41141 C23DKS 11516307 IC50 > 10000 nM T41141 CDA9F5 11517167 Ki > 150000 nM T41141 C6D2VI 11525733 Ki = 2000 nM T41141 CW4ED1 11532268 IC50 = 120 nM T41141 CQ69XF 11533114 Ki = 12000 nM T41141 C2BT3L 11533910 Ki > 150000 nM T41141 C98EQF 11545899 IC50 = 540 nM T41141 C6XK8V 11547772 Ki = 8900 nM T41141 CG57TI 11551229 Ki > 150000 nM T41141 CXTQ39 11558838 Ki = 88000 nM T41141 CF9DE7 11561418 Ki = 71000 nM T41141 CA61ZJ 11562424 Ki = 11000 nM T41141 CKH13D 11562461 Ki = 9100 nM T41141 CTN57Q 11562607 Ki = 1600 nM T41141 CB3W8O 11565199 Ki = 1540 nM T41141 CPY84F 11569750 Ki = 430 nM T41141 CW1O0M 11569883 Ki = 1200 nM T41141 C1TV6S 11580329 Ki = 25000 nM T41141 C73VCU 11584899 Ki = 1.7 nM T41141 CJG6T3 11585276 Ki = 0.57 nM T41141 CER65Q 11588182 Ki = 430 nM T41141 CUX70T 11588744 Ki > 150000 nM T41141 C2Y6JE 11590993 Ki = 2300 nM T41141 CLV84W 11594784 Ki > 150000 nM T41141 C1QO2C 11598043 IC50 = 180 nM T41141 C85WBA 11599792 Ki = 400 nM T41141 CQZ5T4 11602113 Ki > 5000 nM T41141 C1NV2U 11605163 Ki = 11000 nM T41141 CM4OS2 11606272 Ki = 1.4 nM T41141 C98KMP 11612451 Ki = 2200 nM T41141 CZU5E4 11613136 Ki = 8800 nM T41141 CK0AN9 11616537 Ki = 18000 nM T41141 CE8WO5 11618337 Ki = 3200 nM T41141 CTL1P3 11618795 Ki = 420 nM T41141 CQ7KD1 11623853 Ki = 23000 nM T41141 C9LBF3 11628054 Ki = 160 nM T41141 CUS5Q4 11630803 Ki = 45000 nM T41141 C70VTY 11631953 Ki = 7900 nM T41141 C98QKS 11635243 Ki = 7.9 nM T41141 CLMY50 11641509 Ki = 7600 nM T41141 CILB73 11649751 Ki > 17000 nM T41141 CJRN14 11655672 Ki = 15000 nM T41141 C5ZOM0 11656060 IC50 = 16 nM T41141 C0Q7AH 11662896 Ki = 5600 nM T41141 C4YFI9 11663730 IC50 = 10 nM T41141 C0D7NS 11663810 Ki = 16000 nM T41141 C5SJ9K 11669355 IC50 > 10000 nM T41141 C13TGX 11671560 Ki = 540 nM T41141 CT0OZ8 11673881 Ki = 37000 nM T41141 C1BGL5 11677886 Ki = 6400 nM T41141 C23ZVP 11678241 Ki = 8.2 nM T41141 C27LJY 11678922 Ki = 0.43 nM T41141 CDNH37 11680631 Ki > 150000 nM T41141 C1Q2OT 11682028 Ki = 23000 nM T41141 C6Q8KO 11682184 Ki = 5900 nM T41141 CNB67S 11684874 Ki = 12000 nM T41141 CL4XB1 11685284 Ki = 4.5 nM T41141 C53OYX 11692372 Ki = 0.63 nM T41141 C38REW 11695166 Ki > 150000 nM T41141 CJB3E9 11695584 Ki = 48000 nM T41141 C0OC5V 11696208 Ki = 22000 nM T41141 CHP6U3 11699298 Ki = 15000 nM T41141 C7QIP8 11699507 Ki = 10 nM T41141 CRTS62 11703216 Ki = 290 nM T41141 C5UEI7 11703527 IC50 = 6760 nM T41141 C9X6PV 11703830 Ki = 88 nM T41141 CU57OC 11705307 IC50 = 83.7 nM T41141 C0Y5XV 11705688 Ki = 19000 nM T41141 C5FZ1J 11710873 IC50 = 10000 nM T41141 C26RZY 11717535 Ki = 17000 nM T41141 CDS4P0 11743922 Ki = 17 nM T41141 C0SV2T 11753412 Ki = 1490 nM T41141 CY63BP 11761693 IC50 = 90 nM T41141 C8EZR3 11763189 Ki = 1.7 nM T41141 CGU6I7 11767007 Ki = 1.5 nM T41141 C8D7BS 11771234 IC50 > 10000 nM T41141 CT5B1S 11784942 Ki > 33750 nM T41141 CDJH89 11811557 IC50 = 4641 nM T41141 CZ1YB3 11824245 IC50 > 10000 nM T41141 CRXO59 11857300 IC50 = 132 nM T41141 CDOG76 11857302 IC50 = 249 nM T41141 C5NR3L 11962098 IC50 = 83 nM T41141 C3QN1E 11983275 Ki = 1000 nM T41141 C3JO1P 12262704 IC50 > 50000 nM T41141 CP4H9E 12737307 Ki = 122000 nM T41141 C6JS5Y 13184126 Ki > 100000 nM T41141 C31MCN 13186896 IC50 > 100000 nM T41141 CA78NJ 13386706 Ki = 14000 nM T41141 C9WC6M 14655218 Ki = 230 nM T41141 C0XI2R 15296015 IC50 = 3 nM T41141 CLGV32 15547238 IC50 = 42 nM T41141 C2QO1B 15955412 Ki = 123000 nM T41141 CHC31Q 15985697 IC50 = 667 nM T41141 C9LW6H 15985754 IC50 = 67 nM T41141 CQ5F9T 16045426 IC50 = 0.7 nM T41141 CL38RU 16046125 Ki > 100000 nM T41141 CQ2N8D 16046128 Ki = 3120 nM T41141 CY0FX8 16061496 IC50 = 574 nM T41141 C08XJK 16090559 Ki > 10000 nM T41141 CTIV96 16090560 Ki > 10000 nM T41141 C2QWA9 16090561 Ki > 10000 nM T41141 CJBT92 16090562 Ki > 10000 nM T41141 CU6KB8 16090563 Ki > 15000 nM T41141 CZ9J6G 16108888 IC50 = 0.17 nM T41141 C3KMJ0 16108889 IC50 = 5.1 nM T41141 CM7DA6 16108890 IC50 = 0.34 nM T41141 C0M1KY 16108891 IC50 = 1.2 nM T41141 C63XFT 16108892 IC50 = 3.9 nM T41141 C0LJ8Y 16108893 IC50 = 0.33 nM T41141 C7IQ0W 16108894 IC50 = 0.52 nM T41141 CPN5S2 16108895 IC50 = 0.58 nM T41141 CJ98LN 16108900 IC50 = 1.1 nM T41141 CYT2X8 16108901 IC50 = 0.31 nM T41141 CJRB12 16108902 IC50 = 0.45 nM T41141 C0QAC5 16108903 IC50 > 10 nM T41141 CT65ZO 16108904 IC50 = 0.82 nM T41141 CHKR18 16108905 IC50 = 1.7 nM T41141 CZI27Q 16108906 IC50 = 0.68 nM T41141 C5FUL9 16661369 IC50 = 63060 nM T41141 CUTI57 16661526 IC50 = 55728 nM T41141 C26JIW 16661682 IC50 = 17043 nM T41141 C6XPN4 16664855 IC50 = 22 nM T41141 C8XLP2 16720100 Ki > 15000 nM T41141 C4P8ZV 16720327 Ki = 5190 nM T41141 C7Y6EF 16725315 IC50 = 56 nM T41141 CKA87T 17945762 IC50 = 42 nM T41141 CH4TC1 17968209 IC50 > 1000 nM T41141 C0JBH9 18395047 IC50 = 780 nM T41141 C2XTI9 18395048 IC50 = 91 nM T41141 C7WD4Z 18628647 IC50 = 8391 nM T41141 CR7B9L 18628679 IC50 > 10000 nM T41141 CHA0S3 18628693 IC50 = 2755 nM T41141 CU3NM9 18628717 IC50 > 10000 nM T41141 C71IFZ 18628739 IC50 = 9546 nM T41141 CUSD12 18628799 IC50 = 140 nM T41141 C5ZRU1 19540655 IC50 > 100000 nM T41141 CLM2E4 19959068 IC50 = 37000 nM T41141 CP1A6L 20262575 IC50 = 7200 nM T41141 C8O5CM 20828112 Ki = 28000 nM T41141 C2KBL6 22972497 IC50 > 10000 nM T41141 CD5R3V 22972573 IC50 = 2235 nM T41141 CFY7O6 22988664 Ki = 182000 nM T41141 CKW6Q8 23626706 IC50 = 230 nM T41141 CS0G9W 23631927 IC50 = 7 nM T41141 C0QVL2 23644739 Ki = 20 nM T41141 CM1C8V 23644740 Ki = 380 nM T41141 CM5TI6 23644741 Ki = 5040 nM T41141 CMQ72V 23644742 Ki > 100000 nM T41141 CZPF48 23648277 IC50 = 430 nM T41141 CHU59C 23648278 IC50 = 456 nM T41141 CA74XT 23648279 IC50 > 10000 nM T41141 C2I6RW 23648280 IC50 > 10000 nM T41141 CCJ8M5 23648281 IC50 > 10000 nM T41141 C9C0HK 23648282 IC50 = 911 nM T41141 CC50JD 23648283 IC50 = 1035 nM T41141 CS1VW7 23648284 IC50 = 86 nM T41141 CUQH43 23648285 IC50 = 105 nM T41141 CM52JD 23648286 IC50 = 121 nM T41141 CE09VM 23648287 IC50 > 10000 nM T41141 C1FRI4 23648288 IC50 > 10000 nM T41141 C9RNB7 23648289 IC50 = 22 nM T41141 C4J5MD 23648290 IC50 = 15 nM T41141 CY20DH 23648291 IC50 = 23 nM T41141 CF7O3H 23648292 IC50 = 181 nM T41141 CKI1W5 23648293 IC50 = 114 nM T41141 CN5S3K 23648294 IC50 = 24 nM T41141 CTB69E 23648295 IC50 = 41 nM T41141 C31XJH 23648296 IC50 = 7 nM T41141 C5ECI8 23648297 IC50 > 10000 nM T41141 CB7T3I 23648298 IC50 = 1950 nM T41141 CVF2M6 23648299 IC50 = 34 nM T41141 CRZ56K 23648300 IC50 = 1473 nM T41141 CQ1C8H 23648301 IC50 = 809 nM T41141 CQFD10 23648302 IC50 = 560 nM T41141 CFR23Q 23648303 IC50 = 1480 nM T41141 C0FBS2 23648304 IC50 = 771 nM T41141 C67AYX 23648305 IC50 = 1915 nM T41141 CN6R9M 23648306 IC50 = 314 nM T41141 C85PXH 23648308 IC50 = 2422 nM T41141 CVH82R 23648309 IC50 = 342 nM T41141 COZK65 23648310 Ki = 7 nM T41141 CCF89E 23648311 Ki = 216 nM T41141 CS4NV6 23648312 Ki = 22 nM T41141 CC9S7T 23648313 Ki = 4.6 nM T41141 CCTK94 23648314 Ki = 326 nM T41141 CG29HR 23648315 Ki = 134 nM T41141 CY35VT 23648316 Ki = 3.7 nM T41141 CTX79K 23648317 Ki = 1.4 nM T41141 C8T5FW 23648318 Ki = 1.5 nM T41141 C02UQZ 23648319 Ki = 5 nM T41141 C1QVI4 23648320 Ki = 3.4 nM T41141 CP4SY0 23648321 Ki = 2.8 nM T41141 C9C7JR 23648322 Ki = 9.3 nM T41141 CTY4J2 23648323 Ki = 23 nM T41141 CGJ96H 23648326 Ki = 2991 nM T41141 CSI84Q 23648327 Ki = 4214 nM T41141 C2PD6A 23648328 Ki = 1.1 nM T41141 C37FRY 23648329 Ki = 7.2 nM T41141 C4KU8Q 23648330 Ki = 1.2 nM T41141 C09TQZ 23648331 Ki = 25 nM T41141 CM0AG6 23648332 Ki = 13 nM T41141 C8DJZ7 23648333 Ki = 68 nM T41141 CVH46G 23648334 Ki = 14 nM T41141 C1IRW9 23648335 Ki > 79000 nM T41141 CWG7T3 23648336 Ki = 106 nM T41141 CZN75B 23648337 Ki > 37000 nM T41141 CLZX16 23648338 Ki = 148 nM T41141 C5UDE3 23648339 Ki = 303 nM T41141 C7V6EY 23648340 Ki = 176 nM T41141 CRK1M0 23648341 Ki = 7950 nM T41141 C34VFB 23648342 Ki = 1296 nM T41141 CQUD83 23648343 Ki = 316 nM T41141 C32GYK 23648344 Ki > 6440 nM T41141 CHQ82B 23648345 Ki = 14 nM T41141 CH0XM8 23648346 Ki = 120 nM T41141 C8ZT0W 23648347 Ki = 92 nM T41141 C5T6WQ 23648348 Ki = 62 nM T41141 CKE2C0 23648349 Ki = 88 nM T41141 CUH90V 23648350 Ki = 9200 nM T41141 CCA45G 23648351 Ki = 2 nM T41141 CP10ST 23648352 Ki = 15530 nM T41141 CZRA72 23648353 Ki = 1800 nM T41141 CPTK56 23648354 Ki = 20 nM T41141 C1YMU6 23648355 Ki = 19 nM T41141 C58JSH 23648356 Ki = 42 nM T41141 C5YS0D 23648357 Ki = 3410 nM T41141 CNHA15 23648358 Ki = 1.6 nM T41141 CQVC57 23648359 Ki = 75 nM T41141 C03ZCQ 23648360 Ki > 30000 nM T41141 CM5QI0 23648361 Ki > 100000 nM T41141 C6YRH9 23648362 Ki > 100000 nM T41141 CP6Q2L 23648363 Ki > 100000 nM T41141 C63OZA 23648364 Ki > 100000 nM T41141 COU98B 23648365 Ki = 8860 nM T41141 CK43WQ 23648366 Ki = 197 nM T41141 CKQ0P4 23648367 Ki > 30000 nM T41141 CGSN32 23648368 Ki > 100000 nM T41141 C76JKU 23648369 Ki > 100000 nM T41141 C46RQB 23648370 Ki > 30000 nM T41141 CPC7Z2 23648371 Ki > 30000 nM T41141 C5FJZ6 23648372 Ki > 100000 nM T41141 CL8X1T 23648373 Ki > 100000 nM T41141 CL01QA 23648374 Ki = 5470 nM T41141 CG9N8B 23648375 Ki = 6030 nM T41141 CT98GY 23648376 Ki = 9790 nM T41141 CX6JF9 23648377 Ki > 100000 nM T41141 CJ7N9D 23648378 Ki > 100000 nM T41141 C0GQ4R 23648379 Ki > 30000 nM T41141 CYS7Z2 23648380 Ki > 30000 nM T41141 C6H3DY 23648381 Ki > 100000 nM T41141 CGV2J8 23648382 Ki > 100000 nM T41141 CF0JM1 23648383 Ki > 100000 nM T41141 C5LGJ7 23648384 Ki > 100000 nM T41141 C39FZB 23648385 Ki > 100000 nM T41141 C85STC 23648386 Ki > 100000 nM T41141 CWV98T 23648387 Ki > 100000 nM T41141 CX59EJ 23648388 Ki > 100000 nM T41141 CFNX14 23648389 Ki > 100000 nM T41141 CZC34G 23648390 Ki > 100000 nM T41141 C1FJY7 23648391 Ki = 4970 nM T41141 C9KW2O 23648392 Ki = 45 nM T41141 CI58TU 23648393 Ki = 7940 nM T41141 CB3JX0 23648394 Ki = 582 nM T41141 CYBW67 23648395 Ki = 331 nM T41141 CR1K4V 23648396 Ki = 4790 nM T41141 C1B9GH 23648397 Ki = 594 nM T41141 CF72ZM 23648398 Ki = 2570 nM T41141 C9X3TS 23648399 Ki = 232 nM T41141 CL8RT9 23648400 Ki = 75 nM T41141 CPEW28 23648401 Ki = 125 nM T41141 CT10OV 23648402 Ki = 6 nM T41141 CEC70K 23648403 Ki = 4 nM T41141 CE2QR4 23648404 Ki = 2110 nM T41141 C4F2BY 23648405 Ki > 100000 nM T41141 CX37JK 23648406 Ki > 30000 nM T41141 CD8JP5 23648407 Ki = 14600 nM T41141 CC7HD5 23648408 Ki = 2590 nM T41141 CWGL69 23648409 Ki = 512 nM T41141 CA2DE6 23648410 Ki = 1060 nM T41141 C3VT9K 23648411 Ki = 810 nM T41141 CBR76L 23648414 IC50 = 9900 nM T41141 CZ7ME6 23648415 IC50 = 7700 nM T41141 CVU01O 23648416 IC50 = 1100 nM T41141 C3M5GX 23648417 IC50 = 1400 nM T41141 CG9NQ8 23648418 IC50 > 10000 nM T41141 C2F1MC 23648419 IC50 = 8000 nM T41141 CCZ4J1 23648420 IC50 = 2800 nM T41141 CC2W3A 23648421 IC50 = 1700 nM T41141 C8Z5BC 23648422 IC50 = 1200 nM T41141 CVD5Y6 23648423 IC50 = 330 nM T41141 CL4Q2D 23648424 IC50 < 30 nM T41141 CF0TY4 23648425 IC50 = 190 nM T41141 CX0V8M 23648426 IC50 = 154 nM T41141 CME4Y9 23648427 IC50 = 110 nM T41141 C4AJB0 23648428 IC50 = 660 nM T41141 C7DBS2 23648441 Ki = 513 nM T41141 CWY87K 23648448 IC50 = 110 nM T41141 C1YTO9 23648449 IC50 > 10000 nM T41141 CJO2P4 24776563 IC50 = 6680 nM T41141 CR8L2N 24776564 IC50 = 13550 nM T41141 C3U0QR 24776565 IC50 = 4150 nM T41141 CV9F0D 24776566 IC50 > 30000 nM T41141 COZ5C9 24776567 IC50 = 9620 nM T41141 C28RDA 24776568 IC50 > 30000 nM T41141 C9KHL2 24776569 IC50 = 14860 nM T41141 CA4KQ3 24776683 IC50 = 420 nM T41141 C92NZG 24776926 IC50 = 2530 nM T41141 CN1R6S 24776927 IC50 = 3790 nM T41141 CT06JY 24776928 IC50 = 28440 nM T41141 CHF5Y7 24776929 IC50 > 30000 nM T41141 CO3W9N 24776931 IC50 = 3910 nM T41141 C2Y8JF 24776932 IC50 > 30000 nM T41141 CPBT05 24777048 IC50 = 5060 nM T41141 CM4KX2 24777049 IC50 > 30000 nM T41141 C6ACK9 24777050 IC50 = 17100 nM T41141 CCP4V6 24777300 IC50 = 28910 nM T41141 C8JR9Q 24777301 IC50 = 300 nM T41141 CYMF31 24777302 IC50 = 1820 nM T41141 CA04CB 24777303 IC50 = 300 nM T41141 CJ3N1A 24777429 IC50 = 800 nM T41141 CBI96T 24777430 IC50 = 780 nM T41141 CAF5Y4 24777431 IC50 = 500 nM T41141 CB96XZ 24778049 IC50 = 3300 nM T41141 CK74OH 24778050 IC50 = 23280 nM T41141 CQHR89 24778051 IC50 > 30000 nM T41141 CUG91O 24778054 IC50 = 4000 nM T41141 CF30JZ 24778183 IC50 = 10520 nM T41141 CB50GN 24778184 IC50 = 10520 nM T41141 CUP2D4 24778185 IC50 = 13370 nM T41141 C15VPF 24778187 IC50 = 13550 nM T41141 CFWK93 24778188 IC50 > 30000 nM T41141 CF9WJ1 24778189 IC50 = 17140 nM T41141 CVS50O 24778317 IC50 > 30000 nM T41141 CC4TG6 24778318 IC50 = 8050 nM T41141 CTV8S9 24778319 IC50 = 5860 nM T41141 CYP8K1 24778320 IC50 = 2270 nM T41141 CPT6I2 24778321 IC50 = 10790 nM T41141 CKP1F7 24778322 IC50 > 30000 nM T41141 CB64RJ 24778323 IC50 = 6840 nM T41141 C7U5ZK 24778439 IC50 = 2280 nM T41141 CEP4D9 24778440 IC50 = 1170 nM T41141 CH8YB7 24778441 IC50 = 12940 nM T41141 CYCD75 24778442 IC50 = 26920 nM T41141 CB3K0R 24778443 IC50 > 30000 nM T41141 CQ80SX 24778444 IC50 = 610 nM T41141 CV5P1B 24778445 IC50 > 30000 nM T41141 CMI4L3 24800875 Ki = 21900 nM T41141 CAXQ09 24801230 Ki = 13500 nM T41141 CT1A2Z 24801231 Ki = 7000 nM T41141 CN0VA7 24822701 IC50 = 5400 nM T41141 C2GQ6X 24897809 Ki = 0.9 nM T41141 CZ21HD 24898027 Ki = 0.16 nM T41141 CQU38W 24900755 IC50 = 1270 nM T41141 C2S8VB 24901099 IC50 = 26 nM T41141 CIN28B 24901100 IC50 = 263 nM T41141 CD2EH0 24901101 IC50 = 230 nM T41141 CS7B3F 24901102 IC50 = 5816 nM T41141 CG9H6V 25008106 IC50 > 1000 nM T41141 CK7BR0 25023784 IC50 = 5200 nM T41141 CZH87T 25023785 IC50 = 6800 nM T41141 C2PUY3 25023786 IC50 > 1000 nM T41141 CFQM73 25023787 IC50 > 1000 nM T41141 CTK09I 25023788 IC50 = 2300 nM T41141 CDL98C 25023789 IC50 > 1000 nM T41141 CCP3G0 25023790 IC50 > 2000 nM T41141 CGI0U2 25023791 IC50 = 6200 nM T41141 CO72TX 25027584 IC50 = 280 nM T41141 C8CIY2 25030810 IC50 = 1200 nM T41141 CMS0L3 25052748 IC50 > 1000 nM T41141 C7J3MN 25053851 IC50 > 1000 nM T41141 C43JRI 25066441 IC50 = 10.1 nM T41141 C19GML 25071954 IC50 = 150 nM T41141 CF54QZ 25129041 IC50 > 100000 nM T41141 CDO26T 25129042 IC50 > 7943.28 nM T41141 C57LJM 25129043 IC50 > 10000 nM T41141 C3AT6W 25130088 IC50 > 10000 nM T41141 C1FWI6 25133836 IC50 > 10000 nM T41141 CYV1J6 25133837 IC50 > 10000 nM T41141 CBZK08 25133838 IC50 > 50118.72 nM T41141 CUC8N5 25141405 IC50 > 100000 nM T41141 CP8U3Q 25142042 IC50 > 40000 nM T41141 C3C8YJ 25174148 IC50 = 501.19 nM T41141 C5M1BT 25195691 IC50 = 3162.28 nM T41141 CC7TV3 25204336 IC50 > 10000 nM T41141 C73KLE 25209862 IC50 = 4.67 nM T41141 C9FWJ4 25219913 IC50 = 32850 nM T41141 CJ04ZN 25234563 IC50 = 152 nM T41141 CU59SO 25242431 Ki = 16000 nM T41141 C23JPC 25242432 Ki = 14000 nM T41141 CW9JM2 25256832 IC50 = 2000 nM T41141 C3GC7P 25256833 IC50 = 1400 nM T41141 CXU0P9 26794600 Ki = 64000 nM T41141 CTME03 38864605 IC50 = 3150 nM T41141 C26LPI 38864607 IC50 = 9420 nM T41141 CN80BC 38864634 IC50 = 56510 nM T41141 CE4D9Q 40522013 Ki = 17000 nM T41141 CL96WQ 42633150 IC50 = 5246 nM T41141 CZ5F4C 42633340 IC50 = 711 nM T41141 C5XV0H 42633341 IC50 = 49 nM T41141 CZS24P 42633520 IC50 = 98 nM T41141 CI78XT 42633521 IC50 = 1060 nM T41141 CU6PL7 42633691 IC50 = 1086 nM T41141 CQ9TR8 42633692 IC50 = 966 nM T41141 C6FJW2 42634249 IC50 = 1084 nM T41141 C9EN0G 42634411 IC50 = 426 nM T41141 C2ZXJ7 42634578 IC50 = 631 nM T41141 CI25RJ 42634754 IC50 = 436 nM T41141 CZ6B1F 42635119 IC50 = 121 nM T41141 C5X4WG 42635483 IC50 = 219 nM T41141 CZM36T 42641892 IC50 > 10000 nM T41141 CRYH80 42642459 IC50 > 10000 nM T41141 C3DC4M 42647278 Ki = 0.87 nM T41141 C25ELB 44143088 IC50 = 117.49 nM T41141 CL0M7R 44143089 IC50 = 7943.28 nM T41141 C9QDC0 44143091 IC50 = 562.34 nM T41141 CNM6X8 44218399 IC50 = 625 nM T41141 C8Y9NQ 44219712 IC50 = 1240 nM T41141 CJA68L 44224113 IC50 = 251.19 nM T41141 C2V5ZT 44224114 IC50 = 1258.93 nM T41141 C0U9VJ 44224115 IC50 = 501.19 nM T41141 C0MZ9D 44224116 IC50 = 316.23 nM T41141 CEJ82A 44224117 IC50 = 251.19 nM T41141 C0KL7D 44224118 IC50 = 251.19 nM T41141 CE9S0M 44224119 IC50 = 794.33 nM T41141 CV1W0Z 44224120 IC50 = 79.43 nM T41141 C5LDK7 44224121 IC50 = 79.43 nM T41141 C8UF5Q 44224122 IC50 = 316.23 nM T41141 C9YHC5 44224123 IC50 = 50.12 nM T41141 CA26RI 44224124 IC50 = 251.19 nM T41141 CU0PI2 44224125 IC50 = 398.11 nM T41141 CRL79W 44224126 IC50 = 100 nM T41141 C3T0QO 44224127 IC50 = 19.95 nM T41141 C81EVM 44224128 IC50 = 1258.93 nM T41141 C7IY8P 44224129 IC50 = 501.19 nM T41141 CYG02V 44224130 IC50 = 630.96 nM T41141 CJS1B9 44224131 IC50 = 398.11 nM T41141 CN5O8S 44224132 IC50 = 79.43 nM T41141 C2Q3RP 44224133 IC50 = 63.1 nM T41141 CZX62T 44224134 IC50 = 79.43 nM T41141 CP3YA9 44224135 IC50 = 12.59 nM T41141 CSZH31 44224136 IC50 = 12.59 nM T41141 CZ56BP 44263398 IC50 > 20000 nM T41141 CR38EU 44279051 Ki = 47 nM T41141 C5LJS7 44279083 Ki = 16 nM T41141 C2V7RL 44279437 Ki = 39 nM T41141 CD84XF 44279475 IC50 = 15 nM T41141 C0RQ3V 44279712 IC50 = 2.6 nM T41141 CFJ2Z1 44279771 IC50 = 17 nM T41141 C3IBQ0 44279792 IC50 = 3960 nM T41141 CQ57HR 44279823 IC50 = 163 nM T41141 C5YF0J 44279873 IC50 = 37400 nM T41141 C6ZXK0 44280152 IC50 = 166 nM T41141 CVZ54E 44280172 IC50 = 47 nM T41141 CCPA17 44294490 Ki = 90 nM T41141 C2ZHC1 44295739 IC50 = 5400 nM T41141 CNL8Y4 44302956 IC50 = 130 nM T41141 CAM2S5 44302974 IC50 > 10000 nM T41141 CBYD40 44302975 IC50 = 580 nM T41141 CNA24Z 44303031 IC50 > 10000 nM T41141 C56IEO 44303058 IC50 = 10000 nM T41141 CL4VM1 44303061 IC50 > 10000 nM T41141 CS0P5A 44303274 IC50 > 10000 nM T41141 CXU16T 44303285 IC50 = 6000 nM T41141 CEIH70 44303290 IC50 > 10000 nM T41141 CN21AS 44303309 IC50 > 10000 nM T41141 C24EDH 44303315 IC50 = 10000 nM T41141 CDX5M7 44303318 IC50 = 6900 nM T41141 CRK48P 44303319 IC50 > 10000 nM T41141 CKB9O1 44303324 IC50 = 1300 nM T41141 C0FEJ1 44303335 IC50 < 30 nM T41141 CT49MJ 44303338 IC50 = 150 nM T41141 CMF6W2 44303344 IC50 = 30 nM T41141 CD1HJ5 44303345 IC50 = 580 nM T41141 CL26OE 44303389 IC50 = 90 nM T41141 CN9QY5 44303414 IC50 = 10000 nM T41141 CG3OM8 44304535 Ki = 3400 nM T41141 C0FKB3 44304563 Ki = 140000 nM T41141 CC04TQ 44304591 Ki > 150000 nM T41141 C76OIY 44304610 Ki = 3700 nM T41141 CK8JW5 44304611 Ki > 150000 nM T41141 CZ87NW 44304634 Ki > 150000 nM T41141 COR96D 44304861 Ki = 16000 nM T41141 C9O1VP 44319528 Ki = 12 nM T41141 CH9E6N 44321598 Ki = 30 nM T41141 C6EYQ8 44321883 Ki = 29 nM T41141 CTW41Y 44321884 Ki = 52 nM T41141 CU7J2P 44321946 Ki = 154 nM T41141 CKB02C 44329582 Ki = 6340 nM T41141 CTN34G 44329585 Ki = 130 nM T41141 CR1J6F 44329593 Ki = 3000 nM T41141 C3EHF1 44329596 Ki = 790 nM T41141 C97WPV 44329608 Ki = 760 nM T41141 CY5KH4 44329643 Ki = 16700 nM T41141 CJ5W0G 44332538 Ki = 597 nM T41141 C1KD2V 44332539 Ki = 865 nM T41141 C7XQY2 44332540 Ki = 93 nM T41141 C2FHG7 44332555 Ki = 377 nM T41141 C6QOU0 44332714 Ki = 232 nM T41141 C83QDU 44332915 Ki = 299.4 nM T41141 CNO3T1 44342482 IC50 = 0.74 nM T41141 C1IJW5 44343023 IC50 = 8500 nM T41141 C71JRX 44343028 IC50 = 15 nM T41141 COEK09 44343037 IC50 = 270 nM T41141 C61UIS 44343092 IC50 = 110 nM T41141 CB64RL 44343105 IC50 = 1200 nM T41141 C0TAX2 44345292 Ki = 55 nM T41141 CD9P4K 44345387 Ki > 1000 nM T41141 C8HP5M 44347822 IC50 = 2163 nM T41141 CK0B9C 44347827 IC50 > 10000 nM T41141 CO82ZV 44347993 IC50 > 10000 nM T41141 CLCP51 44348116 IC50 = 919 nM T41141 CFBI42 44348134 IC50 = 5783 nM T41141 CYEI89 44348185 IC50 = 338 nM T41141 C3V0GM 44348957 IC50 > 1000 nM T41141 CFI6N5 44348963 IC50 = 23 nM T41141 CNZ2I9 44353889 IC50 = 2400 nM T41141 C9EOS5 44353924 IC50 > 1000 nM T41141 CG1JP8 44353951 IC50 = 1100 nM T41141 CX1IL0 44353974 IC50 = 220 nM T41141 CQ1F6V 44353976 IC50 = 560 nM T41141 CJA79K 44353977 IC50 > 1000 nM T41141 C3GV4U 44353978 IC50 = 1400 nM T41141 C67ZFU 44353986 IC50 = 2800 nM T41141 CT7JK8 44354015 IC50 = 210 nM T41141 C49VSE 44354016 IC50 = 6100 nM T41141 CAC2Q0 44356377 IC50 = 1.4 nM T41141 CU6KO2 44356379 IC50 = 150 nM T41141 C6JTS1 44356381 IC50 = 4.3 nM T41141 CYK6F4 44356399 IC50 = 0.95 nM T41141 CUJK15 44356612 IC50 = 0.74 nM T41141 CBPJ08 44356625 IC50 = 95 nM T41141 C0DE5P 44356626 IC50 = 0.95 nM T41141 CI9OQ6 44356637 IC50 = 3.1 nM T41141 CRA87Z 44356780 IC50 = 4.5 nM T41141 CH9L1E 44356846 IC50 = 5.3 nM T41141 CKS7I4 44357044 IC50 = 0.97 nM T41141 C35ROP 44357071 IC50 = 2.2 nM T41141 C7DOS2 44366435 Ki > 100000 nM T41141 CA9LC3 44382185 Ki = 9 nM T41141 C5NH3W 44382186 Ki = 1 nM T41141 CZU70X 44382187 Ki = 1 nM T41141 C3M5CT 44382237 Ki = 36 nM T41141 C3W7CI 44382238 Ki = 1 nM T41141 CM9WG5 44382239 Ki = 32 nM T41141 CUEX04 44382949 Ki = 7844 nM T41141 C9UQN0 44383254 Ki > 10000 nM T41141 CU4CB8 44383255 Ki = 4110 nM T41141 C83ART 44383306 Ki = 2 nM T41141 CEUA60 44383413 Ki = 2 nM T41141 CX20UA 44383464 Ki = 230 nM T41141 CP7KW2 44391459 IC50 = 130 nM T41141 C9W3HN 44391474 IC50 = 0.71 nM T41141 CV71WQ 44391475 IC50 = 81 nM T41141 CIG5R6 44393795 IC50 = 458 nM T41141 C78QJO 44394249 Ki = 107000 nM T41141 CQRB69 44394250 Ki = 51000 nM T41141 CTRP74 44394287 IC50 = 3000 nM T41141 CP7X6J 44394353 IC50 = 1200 nM T41141 C79NFU 44394458 IC50 = 3000 nM T41141 C2J6MW 44397423 IC50 = 15000 nM T41141 CRSF50 44397609 IC50 = 37000 nM T41141 CHWX97 44397693 IC50 = 130000 nM T41141 CZC50Y 44398247 IC50 > 10000 nM T41141 CQPM06 44398248 IC50 > 10000 nM T41141 CYJ8Z4 44398353 IC50 = 430 nM T41141 CD73QR 44398649 Ki = 0.79 nM T41141 CHQF16 44398651 Ki = 0.025 nM T41141 C4ALQ9 44398659 Ki = 1500 nM T41141 CGQ20I 44398741 Ki = 0.036 nM T41141 CD18YP 44402055 IC50 = 660 nM T41141 CU8TB9 44402056 IC50 = 2600 nM T41141 CD4TP7 44402158 IC50 = 460 nM T41141 CO6BG2 44402160 IC50 = 1700 nM T41141 C0AJC4 44402175 IC50 = 6800 nM T41141 CX9O2Q 44402263 IC50 = 4400 nM T41141 C89MOT 44402291 IC50 = 1000 nM T41141 CFL9B8 44402952 IC50 = 68 nM T41141 CRZT97 44403028 IC50 > 10000 nM T41141 CW2L5D 44404573 Ki = 673 nM T41141 C39PTS 44404574 Ki = 251 nM T41141 CY5NW9 44405210 Ki = 4000 nM T41141 CP8L2A 44405213 Ki = 7500 nM T41141 CA59MJ 44405279 Ki = 22000 nM T41141 C5GS4Y 44405280 Ki > 150000 nM T41141 CDP93F 44405305 Ki = 14000 nM T41141 C64UAX 44405607 Ki = 6400 nM T41141 CI9P8B 44405608 Ki = 4800 nM T41141 C4ZMP9 44408016 IC50 = 11000 nM T41141 C25RIN 44408049 IC50 = 12 nM T41141 C9IEW7 44409018 Ki = 1754 nM T41141 CKC4P5 44411027 Ki = 6000 nM T41141 C2MDN7 44411237 Ki = 4000 nM T41141 CY4H2I 44411981 Ki = 1300 nM T41141 CNU4T9 44412155 Ki = 1 nM T41141 CYF1B9 44412339 Ki > 150000 nM T41141 C1J6OW 44412340 Ki > 150000 nM T41141 CU49OM 44412341 Ki = 63000 nM T41141 CDK32G 44412349 Ki = 4600 nM T41141 CL82XD 44412354 Ki = 100000 nM T41141 C23ZVR 44412355 Ki = 28000 nM T41141 CV26BC 44412365 Ki = 14000 nM T41141 CX93NW 44412366 Ki = 2100 nM T41141 CZN9T0 44412387 Ki = 160 nM T41141 CY90QW 44412402 Ki = 2900 nM T41141 C1HW8F 44412424 Ki = 2900 nM T41141 CYDJ14 44412436 Ki = 960 nM T41141 CV49GB 44412437 Ki = 150000 nM T41141 CZ5VW2 44412440 Ki = 18000 nM T41141 CZR1O3 44412502 Ki = 130000 nM T41141 CA23SL 44414977 Ki = 2500 nM T41141 C0XB2M 44414978 Ki = 360 nM T41141 CAG5F3 44414992 Ki = 680 nM T41141 C8JL9C 44415006 Ki = 540 nM T41141 CS6X7V 44426055 IC50 = 994 nM T41141 C8IB2W 44426056 IC50 > 100000 nM T41141 CVD7L4 44442257 IC50 = 3389 nM T41141 C3J4DH 44444205 IC50 = 96 nM T41141 CX15UA 44444919 IC50 = 2380 nM T41141 CUXF67 44444920 IC50 = 5830 nM T41141 C1DHA5 44444921 IC50 = 9400 nM T41141 CJWB56 44444922 IC50 = 11780 nM T41141 C0NB8D 44444923 IC50 > 30000 nM T41141 C9P7OQ 44444924 IC50 = 870 nM T41141 CXO56L 44447657 IC50 = 2940 nM T41141 CB6H5U 44447658 IC50 > 10000 nM T41141 C1U6JA 44447659 IC50 = 456 nM T41141 CV3T1A 44447660 IC50 > 10000 nM T41141 CF7AV1 44447661 IC50 = 262 nM T41141 C7HRP2 44447662 IC50 = 2650 nM T41141 C0CZ7P 44447663 IC50 = 472 nM T41141 CAF54M 44447664 IC50 = 110 nM T41141 CC4J7S 44447665 IC50 = 750 nM T41141 C7QW0F 44449893 IC50 = 118 nM T41141 CW30VS 44449926 IC50 = 21 nM T41141 C40EDY 44449928 IC50 = 44 nM T41141 C83KAR 44449929 IC50 = 39 nM T41141 C59IFW 44449957 IC50 = 17 nM T41141 CH7YE8 44449958 IC50 = 11 nM T41141 CTQ3A1 44449959 IC50 = 81 nM T41141 CF59ZH 44449960 IC50 = 7.4 nM T41141 C59OXW 44449989 IC50 = 9.4 nM T41141 C69NRS 44449990 IC50 = 3.6 nM T41141 C3KV1I 44450083 IC50 = 2998 nM T41141 CB38OA 44450114 IC50 = 110 nM T41141 C5RQF1 44450115 IC50 = 201 nM T41141 CZU1L6 44450142 IC50 = 21797 nM T41141 CQ7S0A 44450143 IC50 = 41 nM T41141 CNJ3P7 44450179 IC50 = 115 nM T41141 CL6WZ1 44450271 IC50 = 980 nM T41141 C3B2TR 44450349 IC50 > 1000 nM T41141 C38JBH 44450361 IC50 > 1000 nM T41141 CC0AG3 44452909 Ki = 220 nM T41141 CB8IX2 44452912 Ki = 70 nM T41141 CXJF30 44452936 Ki = 30 nM T41141 CVCJ36 44452938 Ki = 1 nM T41141 C4ZBF6 44452963 Ki = 28000 nM T41141 CWCK10 44452964 Ki = 14000 nM T41141 CF9PC3 44452965 Ki = 100000 nM T41141 CF57UN 44456198 IC50 = 133 nM T41141 CKNS35 44456237 IC50 = 34000 nM T41141 C5I2XF 44457308 Ki = 14000 nM T41141 C7HM2X 44457465 Ki = 10700 nM T41141 C91IOW 44457476 Ki = 6000 nM T41141 C2G7LZ 44457481 Ki = 511 nM T41141 C5I0JY 44457489 Ki = 464 nM T41141 CM14NI 44457496 Ki = 24 nM T41141 C70HBQ 44457499 Ki = 21 nM T41141 COR85M 44457502 Ki = 23 nM T41141 C0O8XF 44457507 Ki = 112 nM T41141 CX49LO 44457510 Ki = 45 nM T41141 CKV1E8 44457511 Ki = 155 nM T41141 CIT48F 44457512 Ki = 460 nM T41141 CTUD83 44457513 Ki = 19 nM T41141 C0B4IO 44457516 Ki = 57500 nM T41141 C8Z4WO 44459967 IC50 = 309.03 nM T41141 C86ORE 44459987 IC50 = 204.17 nM T41141 C9TFJ8 44464926 IC50 = 1258.93 nM T41141 CYO0T1 44465454 IC50 = 39.81 nM T41141 CE83YL 44465721 IC50 = 25.12 nM T41141 CVD48M 44478848 IC50 = 730 nM T41141 CJR45G 44479122 IC50 = 355 nM T41141 C8I9QK 44479381 IC50 = 610 nM T41141 CWS3K7 44479385 IC50 = 240 nM T41141 C2PK4G 44479635 IC50 = 48 nM T41141 CB73NC 44479637 IC50 = 145 nM T41141 CA48JP 44480468 IC50 = 1400 nM T41141 C0ZE3C 44480469 IC50 = 1500 nM T41141 C0G5ET 44480470 IC50 = 700 nM T41141 CH7I8C 44480471 IC50 = 400 nM T41141 CPDQ74 44480723 IC50 = 1900 nM T41141 CPN9C7 44480724 IC50 = 1100 nM T41141 CZ62AB 44480725 IC50 = 900 nM T41141 C8SL0N 44480726 IC50 = 2700 nM T41141 C1ZOM7 44480727 IC50 = 900 nM T41141 CZE95Q 44480728 IC50 = 480 nM T41141 CYBH29 44480974 IC50 = 6000 nM T41141 CA0F2M 44480975 IC50 = 460 nM T41141 CFJ21O 44480976 IC50 = 16000 nM T41141 C94NWI 44480977 IC50 = 1000 nM T41141 CFE2H6 44480978 IC50 = 800 nM T41141 COJ38W 44480979 IC50 = 1500 nM T41141 C45EMI 44481231 IC50 = 800 nM T41141 COL4C2 44481232 IC50 = 1400 nM T41141 CJ1M6E 44481233 IC50 = 1100 nM T41141 C32YDM 44481234 IC50 = 1800 nM T41141 CG1X4W 44481235 IC50 = 1600 nM T41141 CG5YU6 44481236 IC50 = 1300 nM T41141 CUHM64 44481503 IC50 = 800 nM T41141 CBGO51 44481504 IC50 = 840 nM T41141 CT9W2X 44481505 IC50 = 600 nM T41141 C1S0KC 44481506 IC50 = 1600 nM T41141 CRQ32O 44481507 IC50 = 190 nM T41141 C1E6AT 44481508 IC50 = 1800 nM T41141 CCW6N4 44481776 IC50 = 1000 nM T41141 CCOK78 44481777 IC50 = 1100 nM T41141 CK1E7H 44481778 IC50 = 900 nM T41141 CFYP92 44482496 IC50 = 130 nM T41141 C1LWX5 44552274 Ki = 4200 nM T41141 CIP6M8 44552275 Ki = 4100 nM T41141 C8W2LG 44552367 Ki = 39700 nM T41141 CWJV95 44552368 Ki = 7700 nM T41141 CIT5G7 44561891 IC50 > 100000 nM T41141 C90BGR 44561892 IC50 > 100000 nM T41141 C9RGX4 44561893 IC50 > 100000 nM T41141 CU7NP5 44561930 IC50 > 100000 nM T41141 CV21IQ 44561931 IC50 > 100000 nM T41141 CR08WA 44561932 IC50 > 100000 nM T41141 CV1IL5 44565796 IC50 > 10000 nM T41141 CLH74F 44565900 IC50 = 1060 nM T41141 CMIP10 44565901 IC50 = 1000 nM T41141 C70BXJ 44565925 IC50 = 1370 nM T41141 CS6YO0 44566187 IC50 = 0.437 nM T41141 CSF17Z 44566188 IC50 > 100000 nM T41141 CJP3U5 44566195 IC50 = 1.66 nM T41141 CUFJ57 44566196 IC50 = 19820 nM T41141 CI6H7R 44568190 IC50 > 2000 nM T41141 CVX81T 44568191 IC50 > 5000 nM T41141 CJRQ74 44568192 IC50 > 1000 nM T41141 C6ZHA4 44568193 IC50 > 1000 nM T41141 C2X3HJ 44568223 IC50 > 1000 nM T41141 CV54EU 44568306 IC50 > 4000 nM T41141 CDZ03Q 44568307 IC50 > 1000 nM T41141 C6FV7W 44568638 IC50 > 1000 nM T41141 C6U3RB 44568639 IC50 = 370 nM T41141 COJ16S 44568640 IC50 = 320 nM T41141 CVP4Y6 44568641 IC50 > 1000 nM T41141 CZW5K2 44568669 IC50 = 260 nM T41141 CW89JM 44568670 IC50 = 840 nM T41141 C2D9TS 44568671 IC50 > 1000 nM T41141 CU4PO0 44568672 IC50 = 23 nM T41141 CCJ68F 44568673 IC50 = 86 nM T41141 CCIP49 44568714 IC50 = 40 nM T41141 C3HYW8 44568715 IC50 > 1000 nM T41141 CLXN21 44568716 IC50 > 1000 nM T41141 CA86UV 44568718 IC50 > 1000 nM T41141 CU82VX 44568766 IC50 > 1000 nM T41141 CZF5G0 44568767 IC50 > 1000 nM T41141 CVR02S 44568768 IC50 > 1000 nM T41141 C1P3LN 44568769 IC50 = 790 nM T41141 CG74ZL 44568770 IC50 > 1000 nM T41141 COHB20 44570671 Ki = 12000 nM T41141 C35ZYP 44570672 Ki = 64000 nM T41141 C3BHM4 44570673 Ki = 16000 nM T41141 C0OSY2 44570674 Ki = 11000 nM T41141 CF41YI 44570719 Ki = 15000 nM T41141 CY9ZT4 44570833 Ki = 7200 nM T41141 CB3S2D 44570834 Ki = 29000 nM T41141 C8K6PB 44570835 Ki = 2000 nM T41141 CWH9Q0 44570836 Ki = 23000 nM T41141 CA10KC 44570876 Ki = 970 nM T41141 CAUD26 44570877 Ki = 7800 nM T41141 C1XCP6 44570878 Ki = 9500 nM T41141 CN1GT2 44570879 Ki = 2300 nM T41141 CV0KJ4 44570915 Ki = 1100 nM T41141 C14JNH 44570916 Ki = 31000 nM T41141 C1DA8K 44570917 Ki = 14000 nM T41141 C9CMZ2 44570957 Ki = 5900 nM T41141 C37LRT 44570958 Ki = 7800 nM T41141 C31BXW 44570959 Ki = 11000 nM T41141 C5G2KT 44570997 Ki = 8400 nM T41141 CZ1ET3 44570998 Ki = 9100 nM T41141 CSYI14 44570999 Ki = 11000 nM T41141 CK5ZM6 44571085 Ki = 7900 nM T41141 CNP2G3 44571086 Ki = 6800 nM T41141 CX2B3F 44571130 Ki = 8500 nM T41141 CFTE86 44571131 Ki = 13000 nM T41141 C4DV1E 44571132 Ki = 14000 nM T41141 C05LYD 44571173 Ki = 13000 nM T41141 CC5A6D 44571174 Ki = 8700 nM T41141 CHB7Y3 44571175 Ki = 23000 nM T41141 C6XF8B 44571212 Ki = 13000 nM T41141 CG5ZO3 44571213 Ki = 24000 nM T41141 C67UMF 44571214 Ki = 27000 nM T41141 CD6X2Y 44571254 Ki = 9100 nM T41141 CQ0W5J 44571255 Ki = 17000 nM T41141 CGM30J 44571297 Ki = 10000 nM T41141 CU0D3P 44571298 Ki = 12000 nM T41141 CUG72S 44571323 Ki = 2500 nM T41141 C2NT4H 44571324 Ki = 11000 nM T41141 CC12QS 44571325 Ki = 27000 nM T41141 CI39YN 44571326 Ki = 15000 nM T41141 C1L3KX 44571358 Ki = 17000 nM T41141 C0NFJ8 44571359 Ki = 21000 nM T41141 CE2PQ4 44571360 Ki = 15000 nM T41141 C5S6FJ 44571361 Ki = 15000 nM T41141 C8YPA6 44572419 Ki = 7400 nM T41141 C3L7IV 44572420 Ki = 2700 nM T41141 CFZ3L7 44572422 Ki = 1900 nM T41141 CFZB79 44572423 Ki = 8400 nM T41141 CGC0W5 44572424 Ki = 3200 nM T41141 C9E6QP 44579079 IC50 = 426 nM T41141 C7CKG9 44579080 IC50 = 276 nM T41141 CFN0Z1 44579081 IC50 > 1000 nM T41141 CH5B0N 44579120 IC50 = 440 nM T41141 CN42GY 44579121 IC50 = 360 nM T41141 CDUJ10 44579122 IC50 = 400 nM T41141 CQJ0L6 44579123 IC50 = 330 nM T41141 CO13BP 44579170 IC50 = 300 nM T41141 CP0X4D 44579171 IC50 = 460 nM T41141 CS60PG 44579172 IC50 = 1390 nM T41141 CY2E6M 44579173 IC50 = 2500 nM T41141 CA0OT2 44587365 IC50 = 64 nM T41141 CM35BH 44587366 IC50 = 270 nM T41141 C2AVQ0 44587440 IC50 = 870 nM T41141 CO7TR5 44587827 IC50 > 2000 nM T41141 CL18MT 44587828 IC50 = 2000 nM T41141 C3A4JO 44587829 IC50 = 780 nM T41141 C9HES8 44587858 IC50 > 3000 nM T41141 CA4DK2 44587859 IC50 > 3000 nM T41141 C76PSY 44587860 IC50 > 3000 nM T41141 C6NU0J 44587861 IC50 > 3000 nM T41141 C8C1OM 44587862 IC50 = 840 nM T41141 CERA06 44587897 IC50 = 1500 nM T41141 CI87JG 44587898 IC50 = 480 nM T41141 C2OQE5 44587899 IC50 = 840 nM T41141 CNM2G4 44587937 IC50 = 700 nM T41141 C65NLR 44587938 IC50 = 510 nM T41141 C81ZSB 44587939 IC50 = 100 nM T41141 CX40GW 46226591 Ki = 850 nM T41141 C8HEC4 46226622 Ki = 13600 nM T41141 CELQ42 46226646 Ki = 7000 nM T41141 CA7V4F 46226655 Ki = 2100 nM T41141 C4YAJ7 46228924 IC50 > 10000000 nM T41141 CD1W6B 46232382 IC50 > 10000 nM T41141 CRYZ16 46232383 IC50 > 10000 nM T41141 C60TNV 46232384 IC50 > 10000 nM T41141 C1I8LN 46232385 IC50 = 2460 nM T41141 C4P7CD 46232387 IC50 > 10000 nM T41141 CQN2I7 46232805 IC50 = 30.5 nM T41141 C39QNG 46232806 IC50 = 1610 nM T41141 CFW92U 46232807 IC50 = 2600 nM T41141 CWD0B5 46232808 IC50 > 10000 nM T41141 CPB62W 46232809 IC50 = 250 nM T41141 CU8ZB6 46232845 IC50 = 131 nM T41141 C32ENI 46232846 IC50 = 46.5 nM T41141 CX0O3T 46232848 IC50 = 79.6 nM T41141 C0WJ4R 46232849 IC50 = 327 nM T41141 CU5KA6 46232850 IC50 > 10000 nM T41141 C5W2SX 46232966 IC50 = 521 nM T41141 CEJ0Z8 46232968 IC50 = 83.8 nM T41141 C60SCN 46232969 IC50 = 610 nM T41141 CL6GY7 46232970 IC50 = 59.4 nM T41141 CA9QH7 46232971 IC50 = 415 nM T41141 C8N2YC 46233007 IC50 = 96 nM T41141 C8HR1S 46233008 IC50 = 233 nM T41141 CY84AW 46233009 IC50 = 114 nM T41141 CRS52G 46233010 IC50 = 118 nM T41141 CC64UL 46233011 IC50 = 63.2 nM T41141 C0U9OQ 46233012 IC50 > 10000 nM T41141 CV74LQ 46233041 IC50 = 2220 nM T41141 C1ZG2T 46233042 IC50 > 10000 nM T41141 C6IJO8 46233043 IC50 = 3320 nM T41141 CZ1E0U 46233044 IC50 > 10000 nM T41141 CH29YW 46233045 IC50 > 10000 nM T41141 CO94IL 46233046 IC50 > 10000 nM T41141 COEI67 46233047 IC50 = 4570 nM T41141 CC2N0F 46842579 IC50 > 10000 nM T41141 CV6SW4 46842581 IC50 > 10000 nM T41141 CM2D1G 46842582 IC50 > 10000 nM T41141 CIU1R5 46842626 IC50 > 10000 nM T41141 C37OSC 46842709 IC50 > 10000 nM T41141 C6HD4M 46865101 IC50 > 10000 nM T41141 CC7DG3 46866398 IC50 = 9772 nM T41141 CGT1Z2 46881448 IC50 > 10000 nM T41141 CH9ON3 46881449 IC50 > 10000 nM T41141 CF15KQ 46881450 IC50 > 10000 nM T41141 CN58BG 46882092 IC50 > 10000 nM T41141 CG9X3C 46882094 IC50 > 10000 nM T41141 CZ5KP8 46882095 IC50 > 10000 nM T41141 CPQZ83 46882096 IC50 > 10000 nM T41141 CUI91D 46905615 IC50 = 560 nM T41141 CS4VM8 46945615 IC50 = 22 nM T41141 CFWU08 46946224 IC50 > 25000 nM T41141 CVT40A 46947220 IC50 = 29700 nM T41141 CAFW31 49783666 IC50 > 10000 nM T41141 CJH50R 49797481 IC50 > 100000 nM T41141 CI7P2B 49797571 IC50 = 15500 nM T41141 CI59MV 49797572 IC50 > 50000 nM T41141 C96CKU 49797573 IC50 = 5400 nM T41141 C9LNK5 49798881 Ki > 150000 nM T41141 CE6Z7V 49798882 Ki = 59900 nM T41141 C5CY7U 49798883 Ki = 12000 nM T41141 C3B8FE 49798886 Ki = 12200 nM T41141 C8R6CQ 49798901 Ki = 2700 nM T41141 C7YZV2 49798902 Ki = 76500 nM T41141 CO7I0B 49798903 Ki = 65000 nM T41141 CVT4U3 49798904 Ki > 150000 nM T41141 C3Y6OC 49798905 Ki = 29800 nM T41141 C4NB3R 49834903 IC50 = 4200 nM T41141 CQ3W9J 49834904 IC50 = 4600 nM T41141 CX1WU8 49834905 IC50 = 2600 nM T41141 CA96LF 49834906 IC50 = 16200 nM T41141 CB9MS2 49834907 IC50 = 2700 nM T41141 C74RAF 49834908 IC50 = 4100 nM T41141 CN8E2A 49834971 IC50 = 1900 nM T41141 COG9T6 49834972 IC50 = 15800 nM T41141 CGPM91 49834975 IC50 = 17000 nM T41141 CJ73DH 49835032 IC50 = 33600 nM T41141 C8XR4Q 49835033 IC50 = 4700 nM T41141 CXE51M 49835035 IC50 = 24900 nM T41141 CKRG17 49835144 IC50 > 25000 nM T41141 C9NO4U 49835145 IC50 > 25000 nM T41141 CP4S5A 49835673 IC50 = 11700 nM T41141 CS3HC6 49835674 IC50 = 12200 nM T41141 C8O3UF 49835732 IC50 = 22200 nM T41141 C37RZT 49862146 IC50 > 10000 nM T41141 CJ0HY8 49862186 IC50 > 10000 nM T41141 CKA53W 49862308 IC50 > 10000 nM T41141 C8B2WE 49862309 IC50 > 10000 nM T41141 CR13LF 49862310 IC50 > 10000 nM T41141 C38BJK 49862365 IC50 > 10000 nM T41141 C1Z9VQ 49862366 IC50 > 10000 nM T41141 C6W1UJ 49862367 IC50 > 10000 nM T41141 CIFP19 49862368 IC50 > 10000 nM T41141 CMW23V 49862369 IC50 > 10000 nM T41141 CI4J0A 49862370 IC50 > 10000 nM T41141 C1XBM6 49862420 IC50 > 10000 nM T41141 CKV06S 49862421 IC50 > 10000 nM T41141 CN4GD6 49862422 IC50 > 10000 nM T41141 CA7K8Q 49862423 IC50 > 10000 nM T41141 CS92IZ 49862471 IC50 > 10000 nM T41141 C1NAQ5 49862472 IC50 > 10000 nM T41141 C5OD6J 49862473 IC50 > 10000 nM T41141 CFCH31 49862474 IC50 > 10000 nM T41141 C29OGE 49862475 IC50 > 10000 nM T41141 CVOG15 49865938 Ki > 100000 nM T41141 CRI85M 50898446 IC50 = 150.8 nM T41141 C18RNG 50925386 Ki = 2700 nM T41141 C4I0JY 50925524 IC50 = 42 nM T41141 C01DJG 50993971 Ki = 860 nM T41141 CW9X3R 50993972 Ki = 480 nM T41141 CIC7H1 50993973 Ki = 1.5 nM T41141 C3UB9Y 50993974 Ki = 2.6 nM T41141 CMS13V 50994055 Ki = 0.4 nM T41141 CPT6I5 50994056 Ki = 0.36 nM T41141 CB4X6Y 50994057 Ki = 0.045 nM T41141 CSY4W0 50994058 Ki = 0.39 nM T41141 CQ08HC 50994059 Ki = 1.4 nM T41141 C30WKN 50994060 Ki = 1.1 nM T41141 C8A1GN 50994137 Ki = 2 nM T41141 C6K3EJ 50994138 Ki = 4.4 nM T41141 CN6ZM0 50994139 Ki = 4700 nM T41141 CF7SN9 50994140 Ki = 940 nM T41141 CU7M1P 50994141 Ki > 22000 nM T41141 C4FE0T 50994142 Ki = 0.22 nM T41141 CJ86MG 51031171 IC50 = 30 nM T41141 C8I1YU 51031462 IC50 = 12 nM T41141 CI1H9F 51031463 IC50 = 6.5 nM T41141 CKNC78 51031601 IC50 = 6.5 nM T41141 CS9Z0X 51031602 IC50 = 4.3 nM T41141 C96FHG 51033722 IC50 = 3600 nM T41141 C6JU9I 51347016 Ki = 690 nM T41141 C2C1YQ 51347017 Ki = 33 nM T41141 C4JB5S 52941092 IC50 > 10000 nM T41141 CDC64G 52941172 IC50 > 10000 nM T41141 C7DO0F 52941283 IC50 = 751 nM T41141 CU1TW6 52941414 IC50 = 458 nM T41141 C71VFU 52941469 IC50 = 891 nM T41141 C8BP5L 52941833 IC50 = 814.5 nM T41141 CQ39TK 52941839 IC50 = 931.3 nM T41141 CDO45C 52941841 IC50 > 10000 nM T41141 CW05MV 52942797 IC50 = 141 nM T41141 C9MK7J 52942931 IC50 = 3819 nM T41141 CVO3U2 52943063 IC50 > 10000 nM T41141 C2AV9H 52943244 IC50 > 10000 nM T41141 CYLF86 52943307 IC50 > 10000 nM T41141 CQDG96 52943578 IC50 > 10000 nM T41141 C4TY6S 52943722 IC50 > 10000 nM T41141 CQ6N0I 52943841 IC50 > 10000 nM T41141 C9B6DJ 52944285 Ki = 3.7 nM T41141 C1UP6N 52945298 IC50 > 10000 nM T41141 CF1LS6 52945475 IC50 > 10000 nM T41141 CN6V0H 52945759 IC50 = 9650 nM T41141 CV8L9Z 52945985 IC50 = 379 nM T41141 CLJ83U 52946267 IC50 > 10000 nM T41141 CBD6S0 52946687 IC50 = 369.7 nM T41141 CS2NX6 52946690 IC50 > 10000 nM T41141 CND9C6 52947170 IC50 > 10000 nM T41141 CT28XU 52947761 IC50 = 2628 nM T41141 CI0S1W 52947952 IC50 > 10000 nM T41141 C75SHQ 52948860 IC50 = 479 nM T41141 C56OCA 53317528 IC50 = 630.96 nM T41141 CM60RJ 53317530 IC50 = 12589.25 nM T41141 C5A6IH 53317737 IC50 = 1258.93 nM T41141 C6FEH9 53318816 IC50 > 25118.86 nM T41141 CJAX07 53318817 IC50 = 2511.89 nM T41141 CG5AP6 53318818 IC50 = 3162.28 nM T41141 CJ3PN0 53319501 IC50 > 10000 nM T41141 C7V2DA 53322116 IC50 > 10000 nM T41141 CQ8O1R 53322117 IC50 > 10000 nM T41141 CR1L4Y 53325394 IC50 > 25118.86 nM T41141 CWJB05 53364091 IC50 = 429 nM T41141 CPN6B8 53378493 IC50 = 9000 nM T41141 C1NJ6T 56654510 Ki > 5000 nM T41141 CDAN29 56657787 IC50 = 3.3 nM T41141 CU26MD 56657788 IC50 = 3.9 nM T41141 CD5W7V 56661312 IC50 = 2 nM T41141 CIX1H6 56664780 IC50 = 6.1 nM T41141 C24ZAM 56664781 IC50 = 2 nM T41141 C24PVH 56664782 IC50 = 3.3 nM T41141 C70CMI 56664783 IC50 = 7.1 nM T41141 CCG3S4 56666730 IC50 = 10 nM T41141 CB57PR 56668196 IC50 = 2.2 nM T41141 CK54CF 56670150 IC50 = 0.53 nM T41141 C69ILG 56670151 IC50 = 22.4 nM T41141 CU59KM 56671669 IC50 = 4.5 nM T41141 C46EFG 56675090 IC50 = 2.1 nM T41141 CDN7E0 56675091 IC50 = 2.2 nM T41141 CA2Z0U 56676986 IC50 = 58.5 nM T41141 CX0FH5 56678398 IC50 = 30 nM T41141 C3WEQ5 56678399 IC50 = 1.9 nM T41141 CD67LW 56678400 IC50 = 2.2 nM T41141 C24QMN 56680316 IC50 = 4400 nM T41141 CX8M7Z 56683636 IC50 = 4.8 nM T41141 CK5X0U 57619789 IC50 > 10000 nM T41141 CH3M0B 59543520 IC50 > 25000 nM T41141 CCR9Q8 59543629 IC50 = 8300 nM T41141 C3ESJ1 59543757 IC50 = 6800 nM T41141 CZV45P 59619390 IC50 > 25000 nM T41141 C75LIT 59907274 Ki = 27 nM T41141 CLX2Y4 60148518 Ki = 37000 nM T41141 C0DA6M 60166364 Ki > 40000 nM T41141 C4G1SF 60166365 Ki > 40000 nM T41141 COM7U3 60166366 Ki > 4000 nM T41141 COQ82A 60166367 Ki > 4000 nM T41141 C2Y7EK 60166492 Ki > 4000 nM T41141 C4PHR1 60166493 Ki > 4000 nM T41141 CG4DZ7 60166494 Ki > 4000 nM T41141 C5E2PB 60166495 Ki > 4000 nM T41141 CXD39V 60166496 Ki > 4000 nM T41141 CM8XO5 60166497 Ki > 4000 nM T41141 C7XLR3 60169906 Ki = 200 nM T41141 CA95CZ 60195809 IC50 > 40000 nM T41141 CY3VC4 60195810 IC50 > 100000 nM T41141 CMA8T3 60195811 IC50 > 100000 nM T41141 CVRJ91 60195812 IC50 = 3110 nM T41141 CE6AH0 60195813 IC50 > 40000 nM T41141 C8ILH6 60195902 IC50 > 10000 nM T41141 CX4N2V 60195903 IC50 > 40000 nM T41141 C4PQ6E 60195904 IC50 > 100000 nM T41141 CNUI89 60195905 IC50 > 40000 nM T41141 C23JUZ 60195906 IC50 > 100000 nM T41141 CBY72G 66572720 Ki = 1500 nM T41141 C34GCU 66572722 IC50 = 16000 nM T41141 CHWA75 66572723 IC50 = 8600 nM T41141 C78CAD 66572724 IC50 = 9000 nM T41141 CAF7U2 66572726 Ki = 900 nM T41141 C3V1BY 66572849 IC50 = 1100 nM T41141 C1Q5WX 66572850 IC50 = 13000 nM T41141 CLJ58E 66572851 Ki = 200 nM T41141 C3VLY0 66572852 IC50 = 19300 nM T41141 C4TXD6 66572853 IC50 = 1500 nM T41141 CJOF37 67298501 Ki = 794.33 nM T41141 C6P9GX 68485393 IC50 = 20000 nM T41141 C4JPF2 69924862 IC50 = 1000 nM T41141 CBR31D 69925026 IC50 = 1300 nM T41141 CVJ5F3 69925527 IC50 = 500 nM T41141 CSF35K 70274227 IC50 > 10000 nM T41141 CI0XF8 70274815 IC50 > 100000 nM T41141 CXT5G7 70275845 IC50 > 10000 nM T41141 C5P3BO 70275923 IC50 > 10000 nM T41141 CCG16F 70276365 IC50 > 100000 nM T41141 C0T3LC 70276605 IC50 > 10000 nM T41141 CE1J0O 70276811 IC50 > 100000 nM T41141 C06WFN 70276830 IC50 > 100000 nM T41141 CDQ85E 70276990 IC50 = 10000 nM T41141 CGET13 70278898 IC50 > 10000 nM T41141 C2GT5H 70280758 IC50 > 100000 nM T41141 CI53XU 70281040 IC50 > 10000 nM T41141 CA6DM2 70281073 IC50 > 100000 nM T41141 CS8VR4 70676096 Ki = 1330 nM T41141 CJQX06 70681840 IC50 = 3600 nM T41141 CW8L0K 70682252 IC50 = 1500 nM T41141 C1UIK4 70682253 IC50 = 284 nM T41141 CSW1R7 70682254 IC50 = 256 nM T41141 CY2WE3 70682255 IC50 > 10000 nM T41141 CVHX94 70682256 IC50 > 10000 nM T41141 CNF23Q 70682257 IC50 = 112 nM T41141 CZ84UX 70682584 IC50 > 100000 nM T41141 CR45PO 70683941 IC50 = 26000 nM T41141 CZI74Q 70683995 IC50 = 26000 nM T41141 CADN96 70683996 IC50 > 50000 nM T41141 C8S1DB 70684341 IC50 > 10000 nM T41141 CH7L2N 70684342 IC50 > 10000 nM T41141 CM5C8Q 70686123 Ki = 1900 nM T41141 CN4QX8 70686124 IC50 = 11000 nM T41141 CM2V0E 70686501 IC50 = 2720 nM T41141 CSPH68 70686502 IC50 > 10000 nM T41141 CL9RE3 70686820 IC50 > 100000 nM T41141 C65EDY 70686822 IC50 > 100000 nM T41141 CBV9F6 70688255 IC50 = 7200 nM T41141 C47WPT 70688256 IC50 = 3200 nM T41141 CMW4T8 70688257 IC50 = 5700 nM T41141 CWE9C8 70688597 IC50 = 46 nM T41141 CV20NB 70688598 IC50 > 10000 nM T41141 CJ4FO1 70688599 IC50 = 1117 nM T41141 CIR23C 70688600 IC50 > 10000 nM T41141 C5NMF8 70688601 IC50 > 10000 nM T41141 C5IYR0 70688897 IC50 > 100000 nM T41141 CA1Q0F 70690660 IC50 = 68 nM T41141 CZY5R0 70690661 IC50 > 10000 nM T41141 C2Z8JP 70690662 IC50 > 10000 nM T41141 C73CZT 70690663 IC50 = 6521 nM T41141 C2H1NL 70690664 IC50 = 260 nM T41141 CLE18H 70692439 IC50 = 2500 nM T41141 CAB1L6 70692440 Ki = 1900 nM T41141 C5D8SA 70692441 IC50 > 50000 nM T41141 CE8Q4U 70692809 IC50 = 434 nM T41141 CND37B 70692810 IC50 > 10000 nM T41141 CZOF81 70693115 IC50 > 100000 nM T41141 CMFW03 70693116 IC50 > 100000 nM T41141 C5RSJ0 70693117 IC50 > 100000 nM T41141 C36JBX 70694841 IC50 > 10000 nM T41141 C86ETZ 70694842 IC50 > 10000 nM T41141 CAU9C4 70694843 IC50 = 3650 nM T41141 C4A7HL 70694844 IC50 = 3960 nM T41141 C01IDC 70695171 IC50 > 100000 nM T41141 CGV1W9 70696541 IC50 > 50000 nM T41141 CXY0A7 70696542 IC50 = 18200 nM T41141 C8HEM6 70696892 IC50 = 214 nM T41141 CK5RP0 70696893 IC50 > 10000 nM T41141 C34WHG 70697225 IC50 > 100000 nM T41141 C0H1BV 70788951 IC50 > 250000 nM T41141 CS60PU 71450699 IC50 = 200 nM T41141 CS58YC 71450700 IC50 = 400 nM T41141 C08LGJ 71451733 IC50 > 10000 nM T41141 CI7Z8B 71451734 IC50 > 10000 nM T41141 C2UN6D 71452029 IC50 > 100000 nM T41141 CG8T7Z 71452030 IC50 > 100000 nM T41141 C7RJG8 71453558 IC50 > 10000 nM T41141 C2OGP1 71453559 IC50 > 10000 nM T41141 CDR10X 71453560 IC50 > 10000 nM T41141 CZ6M8U 71454284 IC50 = 600 nM T41141 CP7H6S 71454285 IC50 > 20000 nM T41141 CFUS41 71455276 IC50 > 10000 nM T41141 CUQL74 71455277 IC50 > 10000 nM T41141 C0KUW5 71455278 IC50 > 10000 nM T41141 C7Z0HF 71455279 IC50 > 10000 nM T41141 C78BKL 71455561 IC50 > 100000 nM T41141 C9YJG7 71457065 IC50 > 10000 nM T41141 C3IH8Z 71457841 IC50 = 18000 nM T41141 CCH47M 71458921 IC50 > 10000 nM T41141 CP7MZ5 71458922 IC50 > 10000 nM T41141 CCA46N 71458923 IC50 > 10000 nM T41141 CQT1C2 71458924 IC50 > 10000 nM T41141 CZT23D 71459213 IC50 = 10800 nM T41141 CF69OZ 71459754 IC50 = 50 nM T41141 CDW0I7 71460731 IC50 > 10000 nM T41141 CC87WL 71460732 IC50 > 10000 nM T41141 CL6Y4C 71460733 IC50 > 10000 nM T41141 C7GX8H 71463202 IC50 = 130 nM T41141 CZM3L7 71520324 Ki = 124000 nM T41141 C5YQ6V 71602930 IC50 > 10000 nM T41141 CY7EL9 71602931 IC50 > 10000 nM T41141 CC61PX 71602932 IC50 > 10000 nM T41141 CH5QG3 71602933 IC50 > 10000 nM T41141 COU6R5 71602979 IC50 > 10000 nM T41141 CR6JV1 71602981 IC50 > 10000 nM T41141 CP87FL 71602983 IC50 = 1740 nM T41141 C34RLW 71602984 IC50 > 10000 nM T41141 CL6B0E 71602986 IC50 > 10000 nM T41141 CQ1ZN0 71603042 IC50 = 658 nM T41141 C6SWY5 71603043 IC50 >= 10000 nM T41141 CD0Z4V 71603045 IC50 > 10000 nM T41141 C1YCF7 71603046 IC50 > 10000 nM T41141 C2VH5F 71603047 IC50 > 10000 nM T41141 CQ76CG 71603106 IC50 > 10000 nM T41141 CF9J1B 71603109 IC50 > 10000 nM T41141 CMSE93 71603111 IC50 > 10000 nM T41141 CIU41Z 71603112 IC50 > 10000 nM T41141 C9GMP4 71603168 IC50 = 228 nM T41141 CSI94H 71612693 Ki = 1700 nM T41141 CH65CP 71612694 Ki = 2600 nM T41141 CER82H 71612695 Ki = 120 nM T41141 C3WV1B 71612696 Ki = 1000 nM T41141 CJ71KZ 71612697 Ki = 20000 nM T41141 COZ0E4 71612901 Ki = 9000 nM T41141 CQ3XD4 71612902 Ki = 1000 nM T41141 C4U0TK 71612903 Ki = 2900 nM T41141 CA82UN 71612904 Ki = 2300 nM T41141 CY02ME 71612905 Ki = 2400 nM T41141 C4TG6P 71612906 Ki = 2600 nM T41141 C3PY2W 71613098 Ki = 2700 nM T41141 C7KF1W 71613099 Ki = 6800 nM T41141 CAG6F9 71613100 Ki = 5500 nM T41141 CI0Q7G 71613101 Ki = 5000 nM T41141 CTH19S 71613102 Ki = 4600 nM T41141 CV60XA 71613103 Ki = 6100 nM T41141 C90OHP 71613322 Ki = 7800 nM T41141 CRP54C 71613323 Ki = 3200 nM T41141 C85WJH 71613324 Ki = 2500 nM T41141 C6HK4W 71615678 Ki = 2400 nM T41141 C7CN4G 71615679 Ki = 1800 nM T41141 C8JN2W 71615680 Ki = 1700 nM T41141 CN32FZ 71615681 Ki = 2500 nM T41141 C4XUV9 71615682 Ki = 23000 nM T41141 CNZ0K4 71624621 IC50 = 67510 nM T41141 C9QY7K 71624622 IC50 = 45270 nM T41141 C0S6HT 71624732 IC50 > 100000 nM T41141 C3CRY6 71624733 IC50 = 73220 nM T41141 C37EVT 71624734 IC50 = 39310 nM T41141 C9P1QH 71624735 IC50 = 91170 nM T41141 CNCX24 71624736 IC50 = 4720 nM T41141 CI5T0R 71656572 Ki = 2.4 nM T41141 CAN6X5 71656574 Ki = 10 nM T41141 C4I0VB 71656669 Ki = 3 nM T41141 CH2J8G 71663299 Ki = 13 nM T41141 C63ROI 71717313 Ki = 155000 nM T41141 C0JYT2 71717876 IC50 = 160 nM T41141 COZB76 71720328 IC50 = 300 nM T41141 C05PXN 71720329 IC50 = 130 nM T41141 C0O5NF 71726670 IC50 = 9.85 nM T41141 CW16QR 71738813 IC50 = 8.12 nM T41141 CS31TK 71738883 IC50 = 14.4 nM T41141 CIO7K3 73345851 Ki = 26000 nM T41141 CY1IU2 73345852 Ki = 390 nM T41141 CDQP51 73347119 Ki = 15000 nM T41141 CJQE58 73348851 Ki = 4200 nM T41141 C5XOV2 73348852 Ki = 27000 nM T41141 C31JUR 73348857 Ki = 740 nM T41141 C95BEA 73348858 Ki = 890 nM T41141 CM3PH8 73350210 Ki = 146000 nM T41141 CZN1M9 73350437 Ki = 3500 nM T41141 CMD57T 73350441 Ki = 7000 nM T41141 CBO54W 73351952 Ki = 28000 nM T41141 COC70E 73351953 Ki = 14000 nM T41141 CAYM96 73351955 Ki = 450 nM T41141 CXR1B9 73353408 Ki = 1400 nM T41141 CNQA65 73354924 Ki = 2600 nM T41141 C37HIQ 73354926 Ki = 3100 nM T41141 CJ6CQ1 73356205 Ki = 400 nM T41141 CL37SD 73356439 IC50 > 10000 nM T41141 CYSR74 73356489 Ki = 4200 nM T41141 CW9NU4 73895627 Ki = 27 nM T41141 CIE28G 73895715 IC50 = 1200 nM T41141 CO68XU 73895952 IC50 = 190 nM T41141 CK3U8P 77907483 IC50 = 2200 nM T41141 CR05TU 89809888 IC50 = 654 nM T41141 CHJB16 89886996 IC50 = 56 nM T41141 CIXT20 89888879 IC50 = 23.8 nM T41141 C62SML 90655967 IC50 > 10000 nM T41141 CJ7LT3 90655968 IC50 > 10000 nM T41141 CB61WC 90655969 IC50 > 10000 nM T41141 CIS56R 90663177 Ki = 720 nM T41141 CU71EO 90663180 Ki = 1000 nM T41141 CX37IK 90663181 Ki = 18 nM T41141 CM4GY1 90663406 Ki = 210 nM T41141 CSD0G2 90663407 Ki = 21 nM T41141 C5F0JO 90663408 Ki = 200 nM T41141 CTNU67 90663409 Ki = 490 nM T41141 CX9NC2 90663410 Ki = 270 nM T41141 CV97ET 90663411 Ki = 3900 nM T41141 CJ2V9B 90663412 Ki = 45 nM T41141 CEZ3N7 90663413 Ki = 240 nM T41141 C7SBR9 90663414 Ki = 270 nM T41141 C9KYG2 90663415 Ki = 160 nM T41141 C7PZ8K 90663416 Ki = 16 nM T41141 C89DWE 90663417 Ki = 67 nM T41141 CX9I6Z 90663418 Ki = 19 nM T41141 C9MQ4F 90663419 Ki = 6600 nM T41141 C0FO3U 90663420 Ki = 210 nM T41141 CF29CP 90663422 Ki = 38000 nM T41141 CJH31Z 90665726 Ki = 25100 nM T41141 CX7WG9 90665730 Ki = 29800 nM T41141 CFKB46 90665732 Ki = 13100 nM T41141 CB14DH 90665735 Ki = 820 nM T41141 C0XZH3 90665919 IC50 = 5870 nM T41141 C0HIA4 90665921 IC50 = 4390 nM T41141 C5AIN7 91667613 IC50 > 10000 nM T41141 CH68BZ 91885514 Ki = 720 nM T41141 CRVO29 91885636 Ki = 11000 nM T41141 CGFK60 101201806 IC50 = 25500 nM T41141 CK0AF8 101889645 IC50 > 100000 nM T41141 C7I4XF 101889646 IC50 > 100000 nM T41141 C8E4WS 102323332 IC50 = 29500 nM T41141 CVJF59 118716317 Ki = 573 nM T41141 CA79YF 118716318 Ki = 228 nM T41141 C3Q5BM 118716319 Ki = 185 nM T41141 CI6H0V 118716320 Ki = 1690 nM T41141 CL4ES1 118716560 IC50 > 100000 nM T41141 C5ALU2 118719334 IC50 = 3300 nM T41141 CTE34I 118720232 IC50 > 100000 nM T41141 CSD62B 118720233 IC50 = 100000 nM T41141 C9WF7Q 118720234 IC50 = 5600 nM T41141 C76HIO 118720235 IC50 > 11000 nM T41141 CAT1R6 118720236 IC50 > 100000 nM T41141 CGAF42 118720237 IC50 > 100000 nM T41141 CJ28KZ 118720238 IC50 > 100000 nM T41141 CPH2V9 118720239 IC50 > 100000 nM T41141 CMBG29 118724585 IC50 = 1000 nM T41141 C35TQG 122186479 Ki = 10000 nM T41141 CF0CG5 122186480 Ki = 1200 nM T41141 CV46XN 122194107 IC50 = 1522 nM T41141 CYO0X5 122194108 IC50 > 10000 nM T41141 CW6K0Z 122194109 IC50 = 5117 nM T41141 CO02XD 122194111 IC50 = 10000 nM T41141 CT51QX 122194112 IC50 = 71.6 nM T41141 CYLN40 122194113 IC50 = 10347 nM T41141 CRS8C6 126610725 IC50 > 10000 nM T41141 CN2IE8 126610758 IC50 >= 10000 nM T41141 C2E4BP 126610767 IC50 >= 10000 nM T41141 C2HJS3 126610779 IC50 > 10000 nM T41141 C2ZL3O 126610781 IC50 > 10000 nM T41141 CJV56I 126610782 Ki = 8.4 nM T41141 CMT2B9 127049869 Ki = 1.27 nM T41141 C43APM 127050163 Ki = 2160 nM T41141 C8VKA5 127050164 Ki = 1920 nM T41141 CZ54XC 127050165 Ki = 431 nM T41141 CI2C3V 127050166 Ki = 6300 nM T41141 CY3JP6 127050263 EC50 = 6000 nM T41141 C7V8XZ 127051317 Ki = 6980 nM T41141 CSK16Q 127051318 Ki = 11700 nM T41141 C7YI4M 127051342 Ki = 4300 nM T41141 C6NFU9 127051343 Ki = 609 nM T41141 C6SD7P 127051344 Ki = 707 nM T41141 CY5CV6 127051345 Ki = 1050 nM T41141 C7HX5O 127054405 IC50 = 320 nM T41141 CEC17N 129164665 Ki = 143 nM T41141 CF9WE3 129164666 Ki = 1522 nM T41141 CY4B7Z 129164668 Ki = 15 nM T41141 CF03SH 129164670 Ki = 181 nM T41141 CEG65P 129164672 Ki = 11 nM T41141 CBSX69 129164675 Ki = 1116 nM T41141 CJO2P0 129164678 Ki = 25 nM T41141 CL9RX5 129164679 Ki = 14 nM T41141 C10YQZ 129164681 Ki = 181 nM T41141 COT2J5 129164699 Ki = 4 nM T41141 CSLH25 129164700 Ki = 1473 nM T41141 CAT90Y 129164701 Ki = 353 nM T41141 CSG89A 129164702 Ki = 82 nM T41141 C89OZL 129164715 Ki = 82 nM T41141 CJ7T4Z 129164725 Ki = 81.7 nM T41141 C3Q5VE 129164742 Ki = 112 nM T41141 CUB58Q 129164743 Ki = 266 nM T41141 CBC15M 129164750 Ki = 76 nM T41141 CS85KM 129164773 Ki = 314 nM T41141 CPG69E 129178768 Ki = 93 nM T41141 CK6I7U 129178772 Ki = 64 nM T41141 C94NGL 129178773 Ki = 7 nM T41141 C41ZCQ 129178794 Ki = 78 nM T41141 CD1I3P 129178829 Ki = 1076 nM T41141 C81SHO 129178830 Ki = 8 nM T41141 CV2LA1 129178843 Ki = 467 nM T41141 C8SD2H 134132002 Ki = 280 nM T41141 C2CT4O 134134083 IC50 = 45 nM T41141 C0U6GR 134134734 Ki = 110 nM T41141 CD5NI4 134134799 Ki = 11 nM T41141 CE53MB 134135884 Ki = 2020 nM T41141 CD0UE9 134136855 IC50 = 17 nM T41141 CW3B7G 134137121 Ki = 49 nM T41141 CF8VA4 134138144 IC50 = 17 nM T41141 C4CT5Z 134139989 Ki = 46 nM T41141 CQ8U5W 134141808 IC50 = 113 nM T41141 C3PEW2 134141970 IC50 = 136 nM T41141 CV36BU 134142724 IC50 = 226 nM T41141 C4BXO1 134144535 IC50 = 23 nM T41141 C4HN8V 134148867 Ki = 30 nM T41141 CH98KJ 134154138 Ki = 19.6 nM T41141 C4TS3J 134154893 IC50 = 17 nM T41141 C2UMT4 134157443 Ki = 200 nM T41141 CEU25N 135137860 Ki = 59000 nM T41141 C5DI9L 135285655 Ki = 253 nM T41141 CNEY95 135285657 Ki = 131 nM T41141 CUVL51 135872798 IC50 = 164 nM T41141 CA8Y4C 136002680 IC50 > 10000 nM T41141 CTQY96 136117851 IC50 = 10 nM T41141 CH08TX 136218747 IC50 > 10000 nM T41141 C2DF5Q 136218748 IC50 > 10000 nM T41141 CL46RX 136218749 IC50 = 449 nM T41141 CGR2E9 136218750 IC50 = 338 nM T41141 CRUC19 137028456 IC50 = 340.5 nM T41141 CS9BV2 137631536 Ki = 1.2 nM T41141 CF94BI 137631849 Ki = 443 nM T41141 CXFL83 137632292 Ki = 217 nM T41141 C13NEP 137633621 Ki = 1430 nM T41141 C23MHJ 137633661 Ki > 5100 nM T41141 CIQ6J5 137633888 Ki = 824 nM T41141 C98CSB 137634116 Ki = 4.6 nM T41141 CBH9O3 137634490 Ki = 2790 nM T41141 CNJ09U 137634671 Ki = 2.5 nM T41141 CI52RD 137635205 Ki = 676 nM T41141 C7Y6UT 137635495 Ki = 7.3 nM T41141 CT5X3N 137635933 Ki = 12 nM T41141 CDF39A 137636254 Ki = 123 nM T41141 CLC04W 137636315 Ki = 1105.7 nM T41141 CG6MH5 137636590 Ki = 30 nM T41141 CT39DN 137637025 Ki = 240 nM T41141 C39AXE 137637300 Ki = 2.2 nM T41141 C7RZ4Q 137638604 Ki = 77 nM T41141 C5MF9X 137638638 Ki = 250 nM T41141 CVJU21 137638762 Ki > 5100 nM T41141 C4W7BD 137638856 Ki = 3860 nM T41141 C25QTS 137639741 Ki = 110 nM T41141 CIZ32F 137639823 IC50 > 10000 nM T41141 CW7IU5 137639903 Ki = 1750 nM T41141 CLX0W9 137640185 Ki = 55.7 nM T41141 CF2QB8 137641334 Ki > 20000 nM T41141 CPV52Z 137641366 Ki > 5100 nM T41141 CO28QB 137642402 Ki = 5.8 nM T41141 CQY6I2 137642965 Ki = 3.7 nM T41141 CVXI65 137643204 Ki = 1364.2 nM T41141 C62IJM 137643751 Ki = 997 nM T41141 CQ98DG 137644516 Ki > 5100 nM T41141 CNS6X7 137644585 Ki = 952 nM T41141 CZC96S 137645782 Ki = 6393.3 nM T41141 CKUJ94 137646266 Ki = 91 nM T41141 C9P6IF 137646532 Ki > 5100 nM T41141 C0TUX3 137646586 Ki = 167 nM T41141 CB7Q5U 137646785 Ki = 7.4 nM T41141 C1AXD7 137647008 Ki = 0.61 nM T41141 CU7BJ0 137647125 Ki = 1.2 nM T41141 CM3OP2 137647368 Ki = 5100 nM T41141 C9F0MH 137647486 Ki = 3020 nM T41141 CZK74L 137647856 Ki = 45 nM T41141 C8FS0C 137649214 Ki = 411 nM T41141 C86ZJA 137649575 Ki = 279 nM T41141 CV54KX 137651518 Ki = 3500 nM T41141 CZBU13 137651934 Ki = 0.4 nM T41141 C4SO3J 137652485 Ki = 1800 nM T41141 CGY3U7 137653100 Ki = 77 nM T41141 CS8U7B 137653242 Ki = 25 nM T41141 CD9P4B 137653316 Ki = 1010 nM T41141 CN79HC 137653449 Ki = 15.5 nM T41141 C4WBO2 137654260 Ki = 505 nM T41141 CG75LU 137654285 Ki = 273.5 nM T41141 C48MPO 137655059 Ki = 1020 nM T41141 C5VI1O 137655103 Ki = 40.3 nM T41141 CR7I0L 137655469 Ki > 5100 nM T41141 C5QVE7 137655537 Ki = 3.5 nM T41141 CB1X4P 137656245 Ki = 304 nM T41141 C6RJO9 137656888 Ki = 25 nM T41141 C4F5SL 137658767 Ki = 671 nM T41141 CZA12J 137659286 Ki = 330 nM T41141 CPA9N7 137659410 Ki > 5100 nM T41141 CL2BY4 137659508 Ki = 5.6 nM T41141 C17LXI 137660025 Ki = 2.3 nM T41141 CT9PH8 137660357 IC50 = 8550 nM T41141 C2FGL6 137660813 Ki = 40 nM T41141 CVP27L 137661274 Ki = 358 nM T41141 C6MI1F 137661465 Ki = 41 nM T41141 CU05SB 137662237 Ki = 515 nM T41141 CEW35U 137662313 Ki = 27 nM T41141 C8A2PN 145960387 IC50 = 92 nM T41141 CFD97H 145960437 IC50 = 2500 nM T41141 C2ER0T 145961056 IC50 = 140 nM T41141 CNJ1G2 145961256 IC50 = 86 nM T41141 C2NFQ1 145961390 IC50 = 110 nM T41141 CAGM09 145961698 IC50 = 1200 nM T41141 C5SLU2 145961778 IC50 = 3500 nM T41141 CIUS59 145962186 IC50 = 280 nM T41141 C3LZB4 145962243 IC50 = 15 nM T41141 CXJ82U 145962422 IC50 = 84 nM T41141 CWYS01 145962673 IC50 = 130 nM T41141 CF8E2T 145962685 IC50 = 4100 nM T41141 CLF40P 145962976 IC50 = 42 nM T41141 CS85OZ 145963002 IC50 = 240 nM T41141 CLP70J 145963229 IC50 = 816000 nM T41141 CY83PE 145963309 IC50 = 140 nM T41141 CSMC76 145963498 IC50 = 590 nM T41141 CJ38RF 145963551 IC50 = 77 nM T41141 C75PCG 145963584 IC50 = 93 nM T41141 CMN91X 145963645 IC50 = 48 nM T41141 CO6UD2 145963721 IC50 = 280 nM T41141 CFQ25D 145967499 IC50 = 755 nM T41141 CIVB10 145967715 IC50 = 4 nM T41141 CLI6T0 145967952 IC50 = 2630 nM T41141 CC4AG7 145968405 IC50 > 5000 nM T41141 CDS31M 145968622 IC50 = 492 nM T41141 CA40YU 145969275 IC50 = 635 nM T41141 CB0Y7Z 145969438 IC50 > 5000 nM T41141 C2WCK0 145969450 IC50 = 300 nM T41141 CL7KO9 145969878 IC50 > 5000 nM T41141 C3NAS7 145970030 IC50 > 5000 nM T41141 C8X6JG 145970039 Ki = 195000 nM T41141 C51ZEH 145970706 Ki = 155000 nM T41141 CS08XI 145970918 IC50 > 5000 nM T41141 C9XKW2 145970931 IC50 = 494 nM T41141 CQ3TG0 145979639 Ki = 22000 nM T41141 CXW3F1 145982578 IC50 = 400 nM T41141 CY7XE4 145982644 IC50 = 4600 nM T41141 C56AXR 145982654 IC50 = 62000 nM T41141 CNC48W 145982661 IC50 = 210 nM T41141 CMS4E9 145982820 IC50 = 260 nM T41141 C7S2TX 145983004 IC50 = 500 nM T41141 CU5Z9F 145983387 IC50 = 2450 nM T41141 CWA21O 145983581 IC50 = 14300 nM T41141 C1OEA0 145983615 IC50 = 500 nM T41141 C6JSW3 145983652 IC50 = 50 nM T41141 C7V2ZF 145983823 IC50 = 1300 nM T41141 CV8HP6 145984203 Ki = 5 nM T41141 C3JIQ4 145984217 IC50 = 18000 nM T41141 CT8QM9 145984597 IC50 = 9500 nM T41141 C3LH7B 145984676 IC50 = 10 nM T41141 CUT36M 145984739 IC50 = 13100 nM T41141 CJM6L4 145984752 IC50 = 400 nM T41141 C0BC2Z 145984777 IC50 = 5300 nM T41141 CJK42D 145985003 IC50 = 180 nM T41141 CGC54P 145985016 IC50 = 1400 nM T41141 C8AM0K 145985030 IC50 = 1490 nM T41141 CURI53 145985037 IC50 = 10 nM T41141 C2LB8K 145985094 IC50 = 200 nM T41141 CNT63X 145985191 IC50 = 30 nM T41141 CHCP90 145985556 IC50 > 2000 nM T41141 CX6JT1 145985564 IC50 = 600 nM T41141 CJE7L9 145985615 IC50 = 37000 nM T41141 CL2B3Y 145985677 IC50 = 1300 nM T41141 C9C5YA 145985785 IC50 = 47000 nM T41141 CBK3G5 145985888 IC50 = 90 nM T41141 CQ2RS8 145986120 IC50 = 1600 nM T41141 CM53FT 145986712 Ki = 5 nM T41141 C6OKB9 145987263 IC50 > 5000 nM T41141 CRD65W 145987430 Ki = 30000 nM T41141 COZ6P5 145987960 IC50 = 4275 nM T41141 C7ZCW3 145988622 IC50 = 334 nM T41141 CN6U8D 145988823 Ki = 5000 nM T41141 C9OAK6 145989037 IC50 = 99 nM T41141 C87GKT 145989707 IC50 = 1591 nM T41141 C8NW1T 145990306 Ki = 12000 nM T41141 C5MWT1 145990477 Ki = 2000 nM T41141 CH7WO9 145994261 Ki = 7300 nM T41141 CUAY08 148018738 IC50 = 3000 nM T41141 CQK39B 149491764 IC50 > 10000 nM T41141 C1ZX5D 149494192 IC50 = 3000 nM T41141 CJ2DW5 155510635 Ki = 1000 nM T41141 CKT12D 155510715 Ki = 1900 nM T41141 CK8F2Z 155512199 Ki = 14.8 nM T41141 COR3E2 155513054 Ki = 10.2 nM T41141 CFN98D 155513234 Ki = 453 nM T41141 CF01VN 155514418 Ki = 630.96 nM T41141 CK6AQ2 155514722 Ki = 398.11 nM T41141 C27SKJ 155515029 IC50 = 0.094 nM T41141 C8HP4U 155515082 Ki > 10000 nM T41141 C6L2RD 155515575 Ki = 230 nM T41141 CJ6Z4N 155515766 Ki = 19.95 nM T41141 CWDS96 155516109 Ki = 47 nM T41141 C5U6FM 155517896 IC50 = 1.35 nM T41141 CYL03V 155518363 Ki = 251.19 nM T41141 CKJ9V2 155519071 IC50 = 0.632 nM T41141 CT94JP 155519833 Ki = 125.89 nM T41141 CE76XY 155520224 Ki = 100 nM T41141 CBK28U 155521458 Ki = 158.49 nM T41141 C0EWD4 155522491 Ki = 5.012 nM T41141 CI9YP3 155522753 Ki = 47 nM T41141 CO2Y0C 155523098 Ki = 700 nM T41141 CZ3KD7 155523939 Ki = 90.3 nM T41141 CBN12I 155524050 Ki = 406 nM T41141 CZI5G3 155524425 Ki = 78.2 nM T41141 C6M1FK 155524435 Ki = 1584.89 nM T41141 CC9X2D 155525224 Ki = 251.19 nM T41141 CD7WG5 155525553 IC50 = 6.64 nM T41141 CNLO46 155526163 Ki = 158.3 nM T41141 CL57AH 155526723 Ki = 108.2 nM T41141 CZ0A5X 155527224 Ki = 158.49 nM T41141 C16ZBY 155529633 Ki = 501.19 nM T41141 C87DAI 155530185 Ki = 39.81 nM T41141 CVN4I3 155530380 Ki = 174.8 nM T41141 C0WZD4 155533248 IC50 = 376 nM T41141 C92YHN 155535180 IC50 = 1.31 nM T41141 CZ59GS 155536157 Ki = 25.12 nM T41141 CB4MT7 155537119 IC50 = 1.68 nM T41141 CYA0Q2 155537428 Ki = 1.5 nM T41141 CNMR90 155537964 IC50 = 3.54 nM T41141 CXHT61 155539577 IC50 = 77 nM T41141 CTV4B7 155539870 IC50 = 1.73 nM T41141 CFRP81 155539888 Ki = 1000 nM T41141 C26AMH 155539986 Ki = 5.3 nM T41141 C95CPE 155540752 Ki = 146000 nM T41141 CO3ZF7 155541809 Ki = 880 nM T41141 C47OMS 155542219 Ki = 100 nM T41141 C43ZKT 155544277 IC50 = 3.53 nM T41141 CB94ZI 155544429 IC50 = 3.13 nM T41141 CIZ8A6 155544625 IC50 = 0.79 nM T41141 CQW2L9 155545346 Ki = 1584.89 nM T41141 CY2TK7 155547967 Ki = 1258.93 nM T41141 CXYT09 155551122 Ki = 195 nM T41141 CT7P2Z 155551886 Ki = 251.19 nM T41141 C3TS9N 155552318 Ki = 158.49 nM T41141 CCF86H 155553085 Ki = 4300 nM T41141 C8Z7GU 155553621 Ki = 630.96 nM T41141 CF0X8Z 155554135 Ki = 199.53 nM T41141 C2P9GA 155554760 IC50 = 47 nM T41141 C6O9FK 155556968 Ki = 1100 nM T41141 C2AIC6 155559777 IC50 = 4.15 nM T41141 CPCR48 155561105 Ki = 35 nM T41141 CRO9V2 155561992 IC50 = 1 nM T41141 CA6XR1 155562235 Ki = 251.19 nM T41141 C1N3AJ 155565629 Ki = 63.1 nM T41141 C3Z7UC 155566273 Ki = 0.6 nM T41141 CW30IO 155567009 Ki = 630.96 nM T41141 CFTW36 155567371 Ki = 76 nM T41141 CLOJ91 155567513 Ki = 4.1 nM T41141 CHD79T 44408017 IC50 = 14000 nM T41141 CO0N3S 44408050 IC50 = 3400 nM T41141 C58OLD 44517711 IC50 = 1.995 nM T41141 CT3S1I 44517712 IC50 = 1.259 nM T41141 CFT38D 45267632 IC50 = 15.85 nM T41141 COU83P 45267640 IC50 = 199.53 nM T41141 C1U4IF 45267645 IC50 = 125.89 nM T41141 CDG5S8 45268499 IC50 = 501.19 nM T41141 CV8PZ3 45268510 IC50 > 7943.28 nM T41141 C89ADF 45269361 IC50 = 794.33 nM T41141 C58PZI 45269375 IC50 = 501.19 nM T41141 C5O9EF 45270206 IC50 = 5.012 nM T41141 C07ADH 45270207 IC50 = 3.981 nM T41141 CVGE81 45270212 IC50 = 6.31 nM T41141 C78EXG 45271021 IC50 = 1995.26 nM T41141 C5MBC4 45271038 IC50 = 5.012 nM T41141 C65QLD 45271887 IC50 = 3981.07 nM T41141 CIL8O6 45271888 IC50 = 1584.89 nM T41141 CLFD35 45272742 IC50 = 3162.28 nM T41141 C3WF8S 45272748 IC50 = 3162.28 nM T41141 CQO98K 45272752 IC50 = 1258.93 nM T41141 C9A0IH 45272753 IC50 = 15.85 nM T41141 CSYU09 45273681 IC50 = 1584.89 nM T41141 C0HRW4 70690665 IC50 > 10000 nM T41141 CU60DG 70696894 IC50 > 10000 nM T41141 D00FGA 73737 IC50 = 1584.89 nM T41141 D00VAN 46232847 IC50 = 224 nM T41141 D01CSE 52942034 IC50 = 232.4 nM T41141 D03JYN 15722900 IC50 = 1020 nM T41141 D04BGT 46881451 IC50 > 10000 nM T41141 D04DFX 136002679 IC50 = 126.1 nM T41141 D05WZF 10129151 IC50 > 5000 nM T41141 D06WQP 60148519 Ki = 15 nM T41141 D08KCA 72429 IC50 = 2.5 nM T41141 D08TMM 9851116 IC50 = 0.2 nM T41141 D08TWJ 10095492 Ki = 970 nM T41141 D09FGQ 123985 IC50 = 13 nM T41141 D09NBP 52940642 IC50 = 1000 nM T41141 D0B2FE 46882093 IC50 > 10000 nM T41141 D0B2JC 46232967 IC50 = 2160 nM T41141 D0B4JS 44449925 IC50 = 910 nM T41141 D0D0JU 14849212 Ki = 10400 nM T41141 D0D0LD 9913088 IC50 = 1221 nM T41141 D0G2QG 44343301 IC50 = 740 nM T41141 D0G8OD 11702208 Ki = 2790 nM T41141 D0J7OM 24777047 IC50 = 4380 nM T41141 D0LL1F 52945875 IC50 = 5410 nM T41141 D0M3AP 46232386 IC50 = 4870 nM T41141 D0MD6D 24778186 IC50 = 12220 nM T41141 D0R2BO 194777 IC50 > 1000 nM T41141 D0S4EI 10244468 Ki = 31700 nM T41141 D0T0IR 49865939 Ki = 3400 nM T41141 D0T7QF 10420833 IC50 = 8900 nM T41141 D0V7LZ 74761 Ki = 11300 nM T41141 D0VE0F 10062714 IC50 = 2000 nM T41141 D0X9YD 65036 Ki = 9300 nM T41141 D0Z0PR 9912381 IC50 = 340 nM T58970 D0J9ZR 4477 IC50 > 100000 nM T58970 D0W5HK 216239 IC50 = 109.5 nM T58970 D01IED 11719003 IC50 < 0.3 nM T58970 D02NNV 3038525 IC50 > 5000 nM T58970 D02RJY 11442891 IC50 > 10000 nM T58970 D03HUX 49792852 IC50 > 10000 nM T58970 D03LWG 53235510 IC50 > 10000 nM T58970 D05ADP 160355 IC50 = 14000 nM T58970 D07EHV 44814409 IC50 > 10000 nM T58970 D07HPJ 11476171 IC50 > 10000 nM T58970 D0CY1B 6420138 Ki > 10000 nM T58970 D0E3TC 44259 IC50 < 1 nM T58970 D0K0YC 9826528 IC50 = 25 nM T58970 D0L1GD 58282870 IC50 = 7 nM T58970 D0O0LS 25141092 IC50 > 10000 nM T58970 D0P1CV 46191454 IC50 > 10000 nM T58970 D0Q4IX 71727581 IC50 = 3.1 nM T58970 D0Q9UX 16718576 IC50 > 10000 nM T58970 D03BNU 59604787 IC50 > 10000 nM T58970 D00PWQ 3820 IC50 = 9000 nM T58970 D00QNV 12111409 IC50 = 37000 nM T58970 D06GXM 12111413 IC50 = 51000 nM T58970 D08DNZ 45102739 IC50 > 50000 nM T58970 D0B6VY 12111411 IC50 = 111000 nM T58970 D0W8BL 46868926 IC50 > 50000 nM T58970 D0YK9D 9956119 IC50 > 10000 nM T58970 D00BPA 4592 IC50 = 7000 nM T58970 D09GHB 11548630 IC50 = 5.8 nM T58970 D09ICC 5164 IC50 = 19000 nM T58970 D0T3ME 156422 IC50 = 9200 nM T58970 C8KED5 4713 IC50 = 2800 nM T58970 C5Q7PG 97297 Ki = 530 nM T58970 CB9F1O 447961 Ki > 1000 nM T58970 C1ZG2U 449087 IC50 > 10000 nM T58970 C67XHJ 660706 IC50 = 18300 nM T58970 CLE2A8 1326085 IC50 = 25600 nM T58970 C38WMR 1380762 IC50 = 14300 nM T58970 CW4EA3 1382118 IC50 = 16900 nM T58970 CL4WX2 1387078 IC50 = 8300 nM T58970 CFQK64 1399707 IC50 = 27400 nM T58970 C5F4WM 1473242 Ki = 2300 nM T58970 C2ZP3H 1875110 IC50 = 23700 nM T58970 CLS85J 1912930 IC50 = 5500 nM T58970 C1SVD2 2132479 IC50 = 27000 nM T58970 CAV19R 2360773 IC50 > 10000 nM T58970 CZHL80 2808202 IC50 > 50000 nM T58970 CJWX69 3848929 IC50 > 100000 nM T58970 CL5I2U 5330279 IC50 > 10000 nM T58970 CZ3LK2 5330387 IC50 > 10000 nM T58970 CRU94N 5330388 IC50 > 10000 nM T58970 CDB68F 5330389 IC50 > 10000 nM T58970 C7CX0H 5330390 IC50 > 10000 nM T58970 C8E0XS 5330391 IC50 > 10000 nM T58970 CW1VX9 5330392 IC50 > 10000 nM T58970 CUEZ35 5330437 IC50 > 20000 nM T58970 C4VQ0B 6419426 IC50 = 560 nM T58970 C5AL8S 6445230 EC50 = 0.55 nM T58970 CA32PV 6540289 IC50 > 50000 nM T58970 CG17TN 6914611 IC50 = 910 nM T58970 C7E2QK 6914613 IC50 = 12850 nM T58970 C16VXB 9863538 IC50 > 10000 nM T58970 CK2J3G 9863776 IC50 = 80 nM T58970 C18HKQ 9885748 IC50 = 13000 nM T58970 C2TC1L 9910609 IC50 = 3040 nM T58970 C3EUB4 9911005 IC50 > 30000 nM T58970 C07VNB 9930243 IC50 = 1288 nM T58970 CJO47T 9948405 IC50 > 10000 nM T58970 C2W3AV 9995236 IC50 > 100000 nM T58970 CV8I5X 9999342 IC50 > 10000 nM T58970 CKSG49 10000883 IC50 > 200000 nM T58970 CS5RF6 10001665 IC50 = 137000 nM T58970 CBW7G9 10001666 IC50 > 200000 nM T58970 C36DGP 10021108 IC50 = 9500 nM T58970 CJ0QI7 10136280 IC50 > 200000 nM T58970 CE4J2D 10155901 IC50 = 29000 nM T58970 CBG09E 10156756 IC50 = 52000 nM T58970 CD3JE0 10177964 IC50 = 103000 nM T58970 C37YAR 10178895 IC50 = 88000 nM T58970 CVYD19 10199925 IC50 = 149000 nM T58970 CGOT91 10207821 IC50 > 100000 nM T58970 CI8MW4 10216627 IC50 = 37000 nM T58970 C5TQ7X 10247543 IC50 > 10000 nM T58970 C6U9MD 10247627 IC50 = 24000 nM T58970 CDA68T 10272087 IC50 > 200000 nM T58970 CG7NU4 10273006 IC50 > 200000 nM T58970 C3LK5B 10293288 IC50 = 22000 nM T58970 C98GPA 10317812 IC50 > 200000 nM T58970 CRT0N9 10339935 IC50 > 200000 nM T58970 CW6L0Q 10339936 IC50 = 230000 nM T58970 CQDM68 10407625 IC50 = 80000 nM T58970 C7HBP6 10429593 IC50 > 10000 nM T58970 C95LYF 10457505 IC50 > 30000 nM T58970 C2WQ8M 10473563 IC50 > 10000 nM T58970 CQ3WB5 10475938 IC50 > 200000 nM T58970 CJ4P5T 10905857 IC50 > 30000 nM T58970 C3ZE1P 11064594 IC50 = 539 nM T58970 C2W5RC 11235063 IC50 > 5000 nM T58970 CBOP58 11293798 Ki = 8210 nM T58970 CE8VP2 11361885 IC50 = 280 nM T58970 C26BZX 11362471 Ki > 10000 nM T58970 C43NPS 11373886 IC50 > 10000 nM T58970 CWXB93 11397177 Ki > 10000 nM T58970 CWM18I 11406175 IC50 > 50000 nM T58970 CFOZ52 11407074 IC50 = 380 nM T58970 C1WXC5 11417488 IC50 > 50000 nM T58970 C64IGY 11448608 Ki > 5000 nM T58970 C0H6QS 11495680 IC50 > 10000 nM T58970 CIW9L5 11502867 IC50 > 10000 nM T58970 CK2Q0X 11516978 IC50 > 10000 nM T58970 CPE53F 11526238 IC50 > 10000 nM T58970 C5BM4T 11531799 IC50 > 10000 nM T58970 C53OSD 11532048 IC50 > 10000 nM T58970 CC4QM5 11532676 IC50 > 10000 nM T58970 CTG83F 11539329 Ki = 5800 nM T58970 C01FVM 11546457 IC50 > 10000 nM T58970 CACS26 11561968 Ki > 4000 nM T58970 CNBM81 11562171 IC50 > 10000 nM T58970 CRO96D 11574520 IC50 = 91000 nM T58970 CFS35Q 11581762 IC50 = 35000 nM T58970 CMIL86 11590363 Ki > 8800 nM T58970 C0NV9Y 11596881 IC50 > 10000 nM T58970 C1BLZ5 11620055 IC50 > 10000 nM T58970 C9T6SC 11640926 Ki = 3900 nM T58970 C24GRQ 11661959 IC50 > 10000 nM T58970 CD29WP 11668438 IC50 = 15.9 nM T58970 CS72ED 11682843 IC50 > 10000 nM T58970 CJ9KN7 11683817 IC50 > 10000 nM T58970 CU0E8O 11690457 Ki = 890 nM T58970 CLC53E 11691173 IC50 > 10000 nM T58970 CB0AP2 11705863 Ki > 4000 nM T58970 C1FTX3 11719305 IC50 > 10000 nM T58970 C9JT4S 11847343 IC50 > 10000 nM T58970 C8E4TS 11992146 IC50 = 4600 nM T58970 CP5VT1 12111410 IC50 = 17000 nM T58970 C6WLE4 12111412 IC50 = 67000 nM T58970 CG3LS7 12111414 IC50 = 23000 nM T58970 C3YRU7 15295578 IC50 = 4600 nM T58970 C7N6CQ 15604547 IC50 = 1200 nM T58970 CO3QF7 15951576 IC50 = 210 nM T58970 CBF4X2 15991561 IC50 > 10000 nM T58970 CFPW41 16007116 Ki = 3400 nM T58970 C9TU1O 16046126 IC50 > 1000 nM T58970 CZHJ34 16058637 IC50 = 25000 nM T58970 CKV4G1 16079040 IC50 = 4000 nM T58970 CU56EW 16664858 IC50 > 10000 nM T58970 C36VTW 16718175 IC50 = 20000 nM T58970 C38FDZ 16760660 IC50 > 10 ug.mL-1 T58970 CZ1QC7 16815741 IC50 = 11000 nM T58970 C5PI9J 20784467 IC50 = 50100 nM T58970 CL81VC 21100709 IC50 = 100000 nM T58970 CM2UY0 23647201 IC50 > 50000 nM T58970 CG6D4M 23647319 IC50 > 10000 nM T58970 CY8Z7X 23647330 IC50 > 10000 nM T58970 C4XD8H 23647348 IC50 > 10000 nM T58970 C2JTA3 23647573 IC50 = 27200 nM T58970 CX63TH 24672456 IC50 = 82000 nM T58970 C7YG1N 24759534 IC50 = 12000 nM T58970 C0VZQ5 24765998 IC50 = 170 nM T58970 C2UOE0 24766030 IC50 > 50000 nM T58970 C8Q7SV 24782039 IC50 = 32000 nM T58970 CMAK08 24782040 IC50 = 43000 nM T58970 CCP2M3 24822704 IC50 > 50000 nM T58970 CC9V2Y 24882562 IC50 > 3000 nM T58970 C43HWQ 24883287 IC50 > 10000 nM T58970 C8DA5Q 24883334 IC50 > 10000 nM T58970 CY8L7E 24896769 IC50 > 10000 nM T58970 CLZ23U 24951610 IC50 = 20000 nM T58970 C4EG8R 24993189 IC50 > 10000 nM T58970 C9AT6X 24995104 IC50 = 5 nM T58970 CEY7V4 24996053 IC50 = 300 nM T58970 C65CFR 24996379 IC50 = 5 nM T58970 CLC39F 24996383 IC50 = 20 nM T58970 CYO8A2 24996697 IC50 = 130 nM T58970 C7P8VK 24996698 IC50 = 36 nM T58970 C2YZ0K 24997018 IC50 = 73 nM T58970 C81KXH 24997019 IC50 = 71 nM T58970 C3P0JO 25067308 IC50 > 200000 nM T58970 C2KY1G 25094210 IC50 > 10000 nM T58970 C6BWZ8 25145145 IC50 > 100 nM T58970 C78YWA 25145716 IC50 > 500 nM T58970 CLFM35 25206064 IC50 = 6300 nM T58970 CNG96H 25210579 IC50 > 10000 nM T58970 C4T7YX 25218756 IC50 = 4300 nM T58970 CC71QJ 27666048 IC50 > 100000 nM T58970 C12NYA 43610313 IC50 = 47000 nM T58970 CO42DC 44138048 IC50 > 100000 nM T58970 CL65QV 44138049 IC50 > 100000 nM T58970 CM86PK 44143527 IC50 = 560 nM T58970 CC9SL5 44143531 IC50 = 1900 nM T58970 CGY5K0 44143533 IC50 = 1300 nM T58970 CFP1N7 44143534 IC50 = 1500 nM T58970 CLW80F 44160269 IC50 > 50000 nM T58970 C0VIX4 44219633 Ki > 4000 nM T58970 CK73NR 44219749 IC50 > 50000 nM T58970 C7PRE3 44315929 IC50 = 50000 nM T58970 C1BWO6 44406125 IC50 = 1400 nM T58970 CN4V5P 44406152 IC50 = 5100 nM T58970 CV09DY 44410717 IC50 > 10000 nM T58970 CP3CI1 44410720 IC50 > 10000 nM T58970 C8W7AD 44410723 IC50 > 10000 nM T58970 CAT5X4 44410829 IC50 > 10000 nM T58970 CC6Y5P 44410844 IC50 > 10000 nM T58970 CG34TY 44410851 IC50 > 10000 nM T58970 C41EIA 44410869 IC50 > 10000 nM T58970 CB6AE8 44410948 IC50 > 10000 nM T58970 CXZG12 44410949 IC50 > 10000 nM T58970 CS7IE9 44410953 IC50 > 10000 nM T58970 CA9M4X 44410954 IC50 > 10000 nM T58970 C3SP5H 44410955 IC50 > 10000 nM T58970 C5D6YP 44410956 IC50 > 10000 nM T58970 C5W1VC 44410959 IC50 > 10000 nM T58970 CM1C2G 44410960 IC50 > 10000 nM T58970 CVSI80 44411048 IC50 > 10000 nM T58970 CN72BR 44411161 IC50 > 10000 nM T58970 C4AW0O 44411183 IC50 > 10000 nM T58970 CETQ79 44427518 IC50 = 5000 nM T58970 COPG94 44427519 IC50 > 10000 nM T58970 C2C4SX 44431829 IC50 > 10000 nM T58970 C9Y1ID 44431830 IC50 > 10000 nM T58970 CU20ER 44431831 IC50 > 10000 nM T58970 CL87AX 44431832 IC50 > 10000 nM T58970 CA61VJ 44431833 IC50 > 10000 nM T58970 C1KW0V 44431834 IC50 > 10000 nM T58970 CHP41T 44442415 IC50 = 448 nM T58970 CI26UX 44442416 IC50 = 899 nM T58970 C2W1RN 44442417 IC50 = 824 nM T58970 C4A9FD 44442418 IC50 = 508 nM T58970 CQEM30 44480711 Ki < 2 nM T58970 CK1Q4M 44481490 Ki < 2 nM T58970 C8G3YW 44481491 Ki = 3 nM T58970 C53EDG 44481492 Ki = 4 nM T58970 CN2PO8 44481493 Ki < 2 nM T58970 C4WHX7 44481494 Ki < 2 nM T58970 CRC7Y6 44481495 Ki < 2 nM T58970 C6MCD5 44481764 Ki < 2 nM T58970 CNFT56 44481765 Ki = 13 nM T58970 CRIB07 44481766 Ki = 15 nM T58970 C24AMY 44481768 Ki < 2 nM T58970 C1XA5C 44481769 Ki < 2 nM T58970 C8LN2S 44482036 Ki = 4 nM T58970 CD3YS7 44482037 Ki = 670 nM T58970 C8MEU4 44482038 Ki < 2 nM T58970 CZO5K0 44482039 Ki < 2 nM T58970 CDOZ57 44482040 Ki = 34 nM T58970 CBJ8U7 44482041 Ki = 5 nM T58970 CX5W3P 44482303 Ki = 5 nM T58970 CKS3B9 44482304 Ki < 2 nM T58970 CNZ38Y 44482305 Ki < 2 nM T58970 C1O8SQ 44482306 Ki < 2 nM T58970 CJ56HF 44482307 Ki = 3 nM T58970 CYH6P3 44520205 IC50 = 296 nM T58970 C4WRN5 44541014 IC50 = 50 nM T58970 C3VRO9 44557921 IC50 > 10000 nM T58970 CCL85F 44575073 IC50 > 50000 nM T58970 CJX06P 44575126 IC50 = 35000 nM T58970 CE8FC7 44575127 IC50 > 50000 nM T58970 C28QLM 44605035 IC50 > 50000 nM T58970 C75XHS 44605037 IC50 > 50000 nM T58970 CU3RF1 45139989 IC50 = 212 nM T58970 CQGZ06 45139991 IC50 = 226 nM T58970 CC95PQ 45375865 IC50 > 50000 nM T58970 CEOQ27 45375866 IC50 > 50000 nM T58970 C96BNW 46179972 IC50 > 50000 nM T58970 CY3HW5 46224684 IC50 > 10000 nM T58970 C7ON5A 46233287 IC50 = 622 nM T58970 COTJ39 46863083 IC50 > 30000 nM T58970 CO3P0J 46866604 IC50 < 50000 nM T58970 CW2G7D 46868853 IC50 > 50000 nM T58970 CR57OZ 46868855 IC50 > 5000 nM T58970 CI8YE5 46868856 IC50 = 35100 nM T58970 C94EPL 46868925 IC50 > 50000 nM T58970 C0GU4D 46868930 IC50 > 50000 nM T58970 CEK2I5 46869149 IC50 = 24000 nM T58970 C1VZM6 46869673 IC50 > 50000 nM T58970 CYI69K 46869674 IC50 > 50000 nM T58970 CSL2N6 46869740 IC50 > 50000 nM T58970 C6V9CD 46869741 IC50 > 50000 nM T58970 CZCQ05 46869742 IC50 > 50000 nM T58970 C09GAW 46869745 IC50 > 50000 nM T58970 CVBG98 46869815 IC50 > 5000 nM T58970 CU2D5N 46869816 IC50 > 50000 nM T58970 C8WH7Q 46869817 IC50 > 50000 nM T58970 CFOX43 46869876 IC50 > 5000 nM T58970 CE0CY1 46869877 IC50 > 50000 nM T58970 C2DW6T 46869878 IC50 > 50000 nM T58970 C19DQG 46869879 IC50 > 50000 nM T58970 CR1OH0 46869880 IC50 > 50000 nM T58970 CD1YH9 46869882 IC50 > 50000 nM T58970 CLS29B 46872626 IC50 > 10000 nM T58970 CZ74MG 46872859 IC50 = 9800 nM T58970 CJOM49 46880136 IC50 > 50000 nM T58970 C2O8RZ 46886323 IC50 > 1000 nM T58970 C2B5XF 49765254 IC50 > 10000 nM T58970 CHSF07 49806372 IC50 > 1000 nM T58970 CBS64G 49830252 IC50 = 59000 nM T58970 CS18HZ 49839481 IC50 > 50000 nM T58970 CJZ5A0 49840306 IC50 > 10000 nM T58970 CB0S2P 49842666 IC50 > 100000 nM T58970 CAI20B 49842778 IC50 > 100000 nM T58970 CRA74I 49842779 IC50 > 10000 nM T58970 CF91RS 49843531 IC50 > 10000 nM T58970 C2Y6QS 50938552 IC50 > 10000 nM T58970 CH4FY5 50941455 IC50 > 50000 nM T58970 CBR71Y 50941538 IC50 > 50000 nM T58970 C4BN7W 50941539 IC50 > 50000 nM T58970 CAZQ43 51003133 IC50 > 1000 nM T58970 C9NYP4 51036677 IC50 > 10000 nM T58970 C4WRY3 51037112 IC50 > 10000 nM T58970 CRI28Z 51037948 IC50 > 10000 nM T58970 CXA03W 52920796 IC50 > 100 nM T58970 CG5IK8 52936268 IC50 = 30 nM T58970 CEQN27 52936621 Ki > 2000 nM T58970 CM24LF 52938983 IC50 = 11380 nM T58970 CA6BH5 52941226 IC50 > 50000 nM T58970 CMXC68 52941286 IC50 > 50000 nM T58970 CAC3J5 52942507 IC50 > 50000 nM T58970 CB1UJ7 52944909 IC50 > 50000 nM T58970 CCMX82 52946092 IC50 > 50000 nM T58970 CLU92X 52948565 IC50 > 50000 nM T58970 CDXL70 52948593 IC50 > 50000 nM T58970 CMT75N 52949817 IC50 > 50000 nM T58970 C4NAB3 53236443 IC50 > 100000 nM T58970 C2CT5J 53236670 IC50 = 429 nM T58970 C3M6LV 53236671 IC50 = 191 nM T58970 C5YZB7 53236674 IC50 > 100000 nM T58970 C5W0BJ 53236676 IC50 > 100000 nM T58970 CZ5L6F 53239373 IC50 = 1130 nM T58970 C2WFI8 53239374 IC50 = 742 nM T58970 C0ZHF8 53239375 IC50 = 1720 nM T58970 CD1EQ3 53239587 IC50 = 733 nM T58970 C1BGN8 53239589 IC50 > 100000 nM T58970 C7XBV1 53239590 IC50 > 100000 nM T58970 CD4M8I 53239593 IC50 = 31600 nM T58970 C6OTY5 53251320 IC50 > 30000 nM T58970 CBTX53 53317412 IC50 > 50000 nM T58970 COCN94 53317413 IC50 > 50000 nM T58970 CHC29T 53317414 IC50 > 50000 nM T58970 C82LCE 53317415 IC50 > 50000 nM T58970 CR0DJ1 53317416 IC50 > 50000 nM T58970 CE8OY2 53317913 IC50 > 100 nM T58970 CP7T3N 53318709 IC50 > 50000 nM T58970 C3TAC2 53320021 IC50 > 5000 nM T58970 CZ0BV7 53320342 IC50 > 10000 nM T58970 COPI53 53321333 IC50 > 50000 nM T58970 C0GLS5 53321334 IC50 > 50000 nM T58970 C2V0QU 53321577 IC50 = 14000 nM T58970 COG9J2 53322644 IC50 > 50000 nM T58970 CUR1A6 53322645 IC50 > 50000 nM T58970 C9SHJ0 53323985 IC50 > 50000 nM T58970 C49MDG 53323986 IC50 > 50000 nM T58970 C3AVG0 53323987 IC50 > 50000 nM T58970 C38RXW 53323989 IC50 > 50000 nM T58970 C2W9OA 53324451 IC50 = 6400 nM T58970 C8VPW5 53325283 IC50 > 50000 nM T58970 CA3X2Q 53325284 IC50 > 50000 nM T58970 CIG7X9 53325285 IC50 > 50000 nM T58970 C4A8JK 53325286 IC50 > 50000 nM T58970 CNT50E 53325288 IC50 > 5000 nM T58970 CV7I4O 53326555 IC50 = 22000 nM T58970 C27IBZ 53326556 IC50 > 50000 nM T58970 C5UK3J 53326557 IC50 > 50000 nM T58970 CVJ6K9 53326558 IC50 > 5000 nM T58970 C8NA4L 53384644 IC50 > 30000 nM T58970 CE1ZK6 54759168 IC50 > 10000 nM T58970 C1XS2J 54760383 IC50 > 10000 nM T58970 CE1O3B 56661803 IC50 > 500 nM T58970 C9DO8G 56682210 IC50 > 50000 nM T58970 CT4E8R 56832546 IC50 = 20000 nM T58970 C6O5WH 56951292 IC50 = 44 nM T58970 CVC0N8 57076369 IC50 = 984 nM T58970 C1JLW8 57332840 IC50 = 2020 nM T58970 CD01JZ 57332841 IC50 = 8430 nM T58970 CCFK37 57332844 IC50 = 3130 nM T58970 CK1SR7 57332969 IC50 = 4260 nM T58970 C5TRE2 57332970 IC50 = 3790 nM T58970 C46TJK 57332974 IC50 = 12210 nM T58970 C09ZJY 57333095 IC50 = 16630 nM T58970 CG2T3Y 57391639 IC50 = 23000 nM T58970 C8QG6P 57393383 IC50 = 73000 nM T58970 C8W6IG 57395117 IC50 > 30000 nM T58970 C7XAP1 57402042 IC50 = 77000 nM T58970 CLB38E 57685675 IC50 = 5.5 nM T58970 CN96GA 57685722 IC50 = 36 nM T58970 CDE3H9 57685726 IC50 = 12 nM T58970 CF59SM 57685880 IC50 = 21 nM T58970 C2XE7K 57686211 IC50 > 3000 nM T58970 CRZY38 57686268 IC50 = 5.6 nM T58970 CPVO76 57686351 IC50 = 23 nM T58970 CP2B1Q 57686448 IC50 = 7 nM T58970 CI19SK 57686585 IC50 = 25 nM T58970 C2ZUY5 58282827 IC50 = 1.7 nM T58970 C8MBE7 58282833 IC50 = 27 nM T58970 CPM97W 58946442 IC50 = 2.1 nM T58970 C9PWZ3 58946448 IC50 = 4.8 nM T58970 CMR6I5 58946455 IC50 = 41 nM T58970 CSO6R7 58985112 IC50 = 36 nM T58970 C2K7PO 58985117 IC50 = 15200 nM T58970 C4AS8Y 58985119 IC50 = 50000 nM T58970 C86ZPG 58985120 IC50 = 980 nM T58970 CZO50Q 58985121 IC50 = 2500 nM T58970 CXO7S1 58985138 IC50 = 1000 nM T58970 CEXC90 58985147 IC50 = 19000 nM T58970 C2TO1W 58985167 IC50 = 360 nM T58970 C8T4OU 58985184 IC50 = 150 nM T58970 C9W4UP 58985193 IC50 = 1200 nM T58970 C6BPR2 58985201 IC50 = 50 nM T58970 CO1W4J 58985202 IC50 = 120 nM T58970 CUM5A8 58985206 IC50 = 2500 nM T58970 C6NDS2 58985207 IC50 > 10000 nM T58970 CUM95O 58985209 IC50 = 73 nM T58970 CMP4X7 58985223 IC50 = 2200 nM T58970 CLXE39 58985237 IC50 = 6000 nM T58970 CE0YM9 58985284 IC50 = 700 nM T58970 CX6DZ4 58985287 IC50 = 170 nM T58970 CQIY86 58985295 IC50 = 1650 nM T58970 CV4DA8 58985303 IC50 = 2300 nM T58970 CXJ63M 59603829 IC50 = 18000 nM T58970 CQEU96 59603842 IC50 = 230 nM T58970 COH62U 60097413 IC50 > 2500 nM T58970 C1MR8Q 60097495 IC50 > 2500 nM T58970 C7YPS1 60198399 IC50 = 2 nM T58970 CIG0P8 60198530 IC50 = 1 nM T58970 CR4K5Z 60198532 Ki = 0.4 nM T58970 CGT3K9 60198589 IC50 = 1 nM T58970 CZH43E 60198725 IC50 = 3 nM T58970 CVQO56 63208024 IC50 = 4600 nM T58970 C1HSE0 67035086 IC50 > 10000 nM T58970 CWI6K5 67035106 IC50 > 10000 nM T58970 C38RGB 67035556 IC50 > 10000 nM T58970 CV63UL 67240318 IC50 > 10000 nM T58970 C4BZW9 67513372 IC50 = 22500 nM T58970 C8I7GC 68293638 IC50 > 10000 nM T58970 CD56XK 68293660 IC50 > 10000 nM T58970 C5DGR9 69036886 IC50 = 1826 nM T58970 C1IEJ2 70789254 IC50 = 47000 nM T58970 C8T7ZP 70789255 IC50 = 38000 nM T58970 CH0B8N 70789756 IC50 > 30000 nM T58970 CPNO23 70844968 IC50 = 24 nM T58970 CZ2JE1 71173380 IC50 = 270 nM T58970 CKT60L 71455860 Ki = 7200 nM T58970 CSE6Z5 71463101 EC50 > 20000 nM T58970 CCN01X 71547862 IC50 > 10000 nM T58970 CA3O6K 71552696 IC50 = 2130 nM T58970 C1NPL0 71552941 IC50 = 14190 nM T58970 CA4PS8 71552942 IC50 = 15950 nM T58970 C3UA9C 71553011 IC50 = 30000 nM T58970 CEZ15Y 71553012 IC50 = 30000 nM T58970 CVIA91 71553085 IC50 = 30000 nM T58970 C1TR3O 71553152 IC50 = 30000 nM T58970 CJ8SA9 71554866 IC50 = 5 nM T58970 C3Y1IH 71555090 IC50 = 12 nM T58970 CQ5TM2 71555167 IC50 = 0.2857 nM T58970 CHO7D1 71555244 IC50 = 0.2 nM T58970 C9VGY4 71555247 IC50 = 0.8512 nM T58970 C0F1AU 71555392 IC50 = 2 nM T58970 CT7W8L 71555462 IC50 = 2 nM T58970 CM04ZX 71555465 IC50 = 0.3 nM T58970 C7AW5O 71555466 IC50 = 0.8 nM T58970 C5HK2E 71555534 IC50 = 0.3 nM T58970 C48RKT 71555839 IC50 = 130 nM T58970 CXSI14 71718330 IC50 > 100000 nM T58970 C1TM3P 71720141 IC50 > 100000 nM T58970 CV4HO3 71726759 IC50 = 490 nM T58970 C35NLY 71726760 IC50 = 89 nM T58970 C6NVW2 71726764 IC50 = 240 nM T58970 CIN10C 71727133 Ki = 0.6 nM T58970 C9AT6G 71727256 Ki = 0.2 nM T58970 COI5S0 71727368 IC50 = 0.94 nM T58970 CV2CR0 71727369 IC50 = 5.9 nM T58970 C23PJX 71727693 Ki = 3 nM T58970 CM8FS0 71727814 Ki = 7.5 nM T58970 CWV5E2 71727815 Ki = 2.5 nM T58970 CHUQ53 71727944 Ki = 0.4 nM T58970 C3V7JE 71728075 Ki = 2.3 nM T58970 CVZ8R6 71728185 Ki = 0.6 nM T58970 CWE3K9 71728186 Ki = 0.1 nM T58970 CF3S6M 71728187 Ki = 1.3 nM T58970 CCVA86 71728296 Ki = 1.6 nM T58970 C0HSC8 73346520 Ki = 2230 nM T58970 C8SD9P 73346521 Ki = 13780 nM T58970 CGZ6Y8 73346522 Ki = 9180 nM T58970 C43IPQ 73348006 Ki = 8840 nM T58970 CS9C0W 73351108 Ki = 1890 nM T58970 C27JUH 73352576 Ki = 778 nM T58970 CVP03Z 73352577 Ki = 4890 nM T58970 CDAB86 73354065 Ki = 2090 nM T58970 CK3Z8U 73354066 Ki = 1730 nM T58970 C92DXZ 73354067 Ki = 9780 nM T58970 CCI18Y 73355591 Ki = 501 nM T58970 CRX8A0 73355592 Ki = 3670 nM T58970 CNM46P 73777037 IC50 = 37 nM T58970 C8W2HV 76309526 Ki = 1000000 nM T58970 C6D0LO 76316736 Ki = 1000000 nM T58970 CJ2T9E 76332983 IC50 > 10000 nM T58970 C5V4LN 78160623 Ki = 0.4 nM T58970 C06ZBG 78160675 Ki = 0.1 nM T58970 CLSY35 78160676 Ki = 1.3 nM T58970 C5PQM0 78160678 Ki = 3.3 nM T58970 C8OU2I 78160679 Ki = 41 nM T58970 CQS1Y8 78160782 Ki = 0.2 nM T58970 CQ2X7Y 78160884 Ki = 6.8 nM T58970 CMZ0T1 78160931 Ki = 2.4 nM T58970 CI0V1O 78160979 Ki = 0.2 nM T58970 CT8G5J 78160981 Ki = 0.5 nM T58970 C29JVD 78160984 Ki = 0.1 nM T58970 CXA9N7 79557014 IC50 = 3200 nM T58970 CHOF41 84973097 Ki = 2.2 nM T58970 CE0RG4 84973098 Ki = 1.7 nM T58970 CGNZ20 84973100 Ki = 0.3 nM T58970 C6ZSG5 84973107 IC50 = 13 nM T58970 C5VA2J 84973109 IC50 = 7.7 nM T58970 C8VP5N 86298673 Ki = 0.6 nM T58970 CPG3A5 86302574 IC50 > 30000 nM T58970 CP0WM3 86696674 IC50 = 4.1 nM T58970 CTD4J1 86696703 Ki = 1.1 nM T58970 CA49FO 86705475 IC50 = 17 nM T58970 CS1DU0 89536143 IC50 = 0.9 nM T58970 C1HW4B 89735655 IC50 = 1200 nM T58970 COA52P 89784628 Ki = 0.6 nM T58970 C1O0BS 89794860 IC50 = 37 nM T58970 C6BPV7 89794862 Ki = 2.8 nM T58970 CL23IO 89794863 Ki = 0.5 nM T58970 CM6S7U 89794864 Ki = 0.3 nM T58970 CV84CW 89794964 Ki = 2.4 nM T58970 CWPU14 89794970 Ki = 6.8 nM T58970 CI32KM 89795018 Ki = 1.5 nM T58970 C1VD2Z 89795025 Ki = 0.1 nM T58970 C54NBM 89795059 IC50 = 17 nM T58970 CYLX17 89795073 IC50 = 29 nM T58970 CZVQ60 89795088 Ki = 1.5 nM T58970 CO1UM8 89795095 IC50 = 5650 nM T58970 CSI76W 89795096 Ki = 0.3 nM T58970 CC58FK 89795228 Ki = 1.5 nM T58970 CP3D0E 89795229 Ki = 1.2 nM T58970 CPHT17 89795256 IC50 = 10 nM T58970 C6KBW4 89795275 IC50 = 16 nM T58970 CW5O1N 89795280 IC50 = 290 nM T58970 C15FCX 89795282 IC50 = 52 nM T58970 CN4VB6 89795308 IC50 = 0.9 nM T58970 C1MEH3 89795309 Ki = 1.8 nM T58970 C3A2KY 89795319 Ki = 0.8 nM T58970 C49SCO 89795321 Ki = 0.4 nM T58970 CU3SJ4 89795322 Ki = 0.3 nM T58970 CH96XR 89807408 Ki = 1.8 nM T58970 CSK8C3 89807688 IC50 = 1.8 nM T58970 COG5U9 89807745 Ki = 0.7 nM T58970 C6GME9 89807821 IC50 = 23 nM T58970 CJVM86 89807905 Ki = 14 nM T58970 C81OIU 89807999 Ki = 0.4 nM T58970 C2OAR8 90104994 IC50 = 280 nM T58970 CP81ZY 90105293 IC50 = 5900 nM T58970 C9R8IF 90105361 IC50 = 11700 nM T58970 CBPE29 90105453 IC50 = 72 nM T58970 CJN63K 90105551 IC50 = 252 nM T58970 CMGA83 90105804 IC50 = 634 nM T58970 CDP72E 90105816 IC50 = 354 nM T58970 CDIA15 90105999 IC50 = 416 nM T58970 CM7L3B 90106032 IC50 = 71 nM T58970 C06RPO 90106116 IC50 = 149 nM T58970 C6PHF1 90331409 IC50 = 5.4 nM T58970 CY0UC4 90645194 IC50 > 10000 nM T58970 CXV2R0 90645247 IC50 = 4 nM T58970 C90SKQ 90645248 IC50 = 2 nM T58970 CXZ0H7 90645249 IC50 = 21 nM T58970 C1Z6GR 90645250 IC50 = 51 nM T58970 C3CGL5 90645251 IC50 = 3 nM T58970 C8BPR2 90645252 IC50 = 2 nM T58970 C8FOU6 90645255 IC50 = 2 nM T58970 CDWB05 90645256 IC50 = 12 nM T58970 CYI9F1 90645257 IC50 = 106 nM T58970 C5A1QM 90645258 IC50 = 283 nM T58970 CJC39W 90645259 IC50 = 69 nM T58970 C02NTP 90645260 IC50 = 91 nM T58970 C52BPM 90645261 IC50 = 93 nM T58970 C2S9XB 90645262 IC50 = 1856 nM T58970 CE5LY0 90645263 IC50 = 81 nM T58970 C6ZP2X 90645264 IC50 = 66 nM T58970 CXIS31 90645265 IC50 = 4 nM T58970 C62FNS 90645266 IC50 = 6 nM T58970 C3TN0C 90645267 IC50 = 2 nM T58970 CY6F8O 90645268 IC50 = 11 nM T58970 CKMH46 90645269 IC50 = 122 nM T58970 C3JM9Q 90645270 IC50 = 356 nM T58970 CD94KZ 90645271 IC50 = 4 nM T58970 CNLO67 90645272 IC50 = 8 nM T58970 C8B1VE 90645273 IC50 = 7 nM T58970 C8XW0Z 90645274 IC50 = 43 nM T58970 C95MOT 90645275 IC50 = 20 nM T58970 C4TQ3S 90645276 IC50 = 9 nM T58970 CSR85G 90645277 IC50 = 4 nM T58970 C0R6OK 90645279 IC50 = 41 nM T58970 C1A3ZX 90645280 IC50 = 2 nM T58970 C76IFU 90645281 IC50 = 348 nM T58970 C75SQL 90645282 IC50 = 26 nM T58970 C34JDS 90645284 IC50 = 93 nM T58970 CJ6D0P 90645285 IC50 = 6 nM T58970 C91KIJ 90645286 IC50 = 7 nM T58970 C65ANP 91666625 IC50 = 0.19 nM T58970 C8S2XK 91758407 IC50 = 260 nM T58970 CG2Y7L 91809196 IC50 = 6.9 nM T58970 CU51BA 91819624 IC50 = 3 nM T58970 C05UCQ 91819625 IC50 = 89 nM T58970 C5Q3AE 91819626 IC50 = 5 nM T58970 C39YGT 91864560 IC50 = 0.16 nM T58970 C6N3JK 91864561 IC50 = 0.01 nM T58970 C46MDT 91864562 IC50 = 0.19 nM T58970 CAU45T 91971978 IC50 > 30000 nM T58970 C78ZDC 92044553 IC50 = 0.9 nM T58970 CYMH49 92044895 IC50 = 0.3 nM T58970 CY61QP 92044904 IC50 = 4 nM T58970 C2P3LF 102136592 IC50 = 1600 nM T58970 CL64EZ 102287891 IC50 > 10000 nM T58970 C2NQ4S 102287892 IC50 > 10000 nM T58970 CZG9I3 118030039 IC50 = 1 nM T58970 CG1A0F 118275149 IC50 = 468 nM T58970 CA17JS 118275156 IC50 = 623 nM T58970 C26JBO 118369772 IC50 = 10 nM T58970 CY7BI2 118706214 IC50 > 10000 nM T58970 C3Y9WQ 118721299 IC50 = 930 nM T58970 C0NE8X 118721300 IC50 = 440 nM T58970 CF3SX2 118721301 IC50 = 280 nM T58970 C2J1NV 118722546 IC50 = 3 nM T58970 C8Y5MR 118727592 IC50 = 71 nM T58970 CQCX41 118737057 IC50 > 10000 nM T58970 CH56TP 121416353 IC50 = 733.9 nM T58970 CIHB61 121416358 IC50 = 5.014 nM T58970 CYCV06 121416382 IC50 = 757.3 nM T58970 CO1IK8 121416413 IC50 = 16.22 nM T58970 CCQ8G3 121416421 IC50 = 8.791 nM T58970 CV6T5C 121416436 IC50 = 10.22 nM T58970 CW12TI 121428523 IC50 = 0.9958 nM T58970 C63TGL 121428526 IC50 = 6.284 nM T58970 CSN73I 121428528 IC50 = 5.088 nM T58970 C7Q2FD 121428532 IC50 = 3.535 nM T58970 CIN0M7 121428533 IC50 = 3.443 nM T58970 CN3Q4R 121428534 IC50 = 13.62 nM T58970 C21HYN 121428535 IC50 = 687.3 nM T58970 CQC6I7 121428539 IC50 = 4.107 nM T58970 C0BAC2 121428620 IC50 = 633.5 nM T58970 CBY4V9 121428621 IC50 = 14.49 nM T58970 C2TSV7 122177851 IC50 = 54 nM T58970 CEK9S7 122177852 IC50 = 44 nM T58970 C40APN 122177853 IC50 = 43 nM T58970 CCN6F5 122177854 IC50 = 3.2 nM T58970 CE68SL 122177855 IC50 = 4.7 nM T58970 CSFJ19 122177913 IC50 = 5.4 nM T58970 C53NSH 122177914 IC50 = 4.3 nM T58970 CJD03F 122177915 IC50 = 5.3 nM T58970 CX8JI0 122177916 IC50 = 3.4 nM T58970 CJI3N8 122177917 IC50 = 4.6 nM T58970 CJHF98 122177918 IC50 = 23 nM T58970 CU15EY 122177919 IC50 = 23 nM T58970 CGDL13 122177920 IC50 = 78 nM T58970 CVE19K 122177921 IC50 = 43 nM T58970 CB1HF0 122177922 IC50 = 89 nM T58970 CER2Y0 122177923 IC50 = 21 nM T58970 COQ7U6 122177924 IC50 = 2.3 nM T58970 CV1A2F 122177925 IC50 = 3.5 nM T58970 CJ6RM1 122177926 IC50 = 7 nM T58970 CC13JY 122177927 IC50 = 4.5 nM T58970 C8GB4Q 122181008 IC50 > 10000 nM T58970 CBQ94Z 122181009 IC50 > 10000 nM T58970 CT8CP2 122181010 IC50 > 10000 nM T58970 CB6IZ0 122181011 IC50 > 10000 nM T58970 C65BOF 122181012 IC50 > 10000 nM T58970 CO83PN 122181013 IC50 > 10000 nM T58970 CE6D5X 122181354 IC50 = 240 nM T58970 C8O7YN 122181355 IC50 = 7.5 nM T58970 C8V5HL 122181356 IC50 = 74 nM T58970 CF5LQ7 122181357 IC50 = 9000 nM T58970 C8GW5V 122181358 IC50 = 1800 nM T58970 CU4ZK1 122181359 IC50 = 380 nM T58970 C9LTM2 122181360 IC50 = 42 nM T58970 CB9GK1 122181361 IC50 = 480 nM T58970 CQ94UG 122181362 IC50 = 3.1 nM T58970 CAS9U2 122181363 IC50 = 170 nM T58970 CSON37 122181364 IC50 = 9.9 nM T58970 CNIA82 122181365 IC50 = 90 nM T58970 CYDH02 122181366 IC50 = 39 nM T58970 CP08YF 122186070 IC50 = 11 nM T58970 C14WSQ 122186071 IC50 = 550 nM T58970 CRJ81U 122186072 IC50 = 7 nM T58970 C1BR8U 122186073 IC50 = 76 nM T58970 CG4OY0 122186074 IC50 = 0.5 nM T58970 C8OK7L 122186075 IC50 = 0.3 nM T58970 CTF36V 122186076 IC50 = 0.2 nM T58970 CMIL75 122186077 IC50 = 0.4 nM T58970 C46YAE 122186078 IC50 = 0.7 nM T58970 CX1Y8T 122186079 IC50 = 1.8 nM T58970 CP3F4S 122186080 IC50 = 4.6 nM T58970 CU7V1S 122186888 IC50 = 0.26 nM T58970 C2ZQ1H 122186889 IC50 = 2.26 nM T58970 C2TML6 122186890 IC50 = 0.033 nM T58970 C5J2IP 122186891 IC50 = 0.04 nM T58970 C2FZ3L 122186892 IC50 = 0.035 nM T58970 C3Z2DE 122186993 IC50 = 0.026 nM T58970 C65QIL 122186994 IC50 = 0.05 nM T58970 CPL41V 122186995 IC50 = 0.019 nM T58970 CDHZ51 122186996 IC50 = 76 nM T58970 C5QIT9 122193281 IC50 > 200000 nM T58970 CYCR35 122193282 IC50 > 200000 nM T58970 CAS9Z1 122193283 IC50 = 44100 nM T58970 C8T4BA 122193284 IC50 = 89700 nM T58970 C2JO7B 122193285 IC50 = 29700 nM T58970 CAM5N1 122193287 IC50 = 21600 nM T58970 C0WVY8 122193401 IC50 = 71500 nM T58970 C76FTO 122193402 IC50 = 14000 nM T58970 C6RKG4 122193403 IC50 = 22200 nM T58970 CRH6M8 122193404 IC50 = 31900 nM T58970 CG16QS 122193405 IC50 = 407 nM T58970 C92XHZ 122193406 IC50 = 2200 nM T58970 C1I2KQ 122193407 IC50 = 1050 nM T58970 CBS38L 122193408 IC50 = 182 nM T58970 CGM9P7 122193409 IC50 = 91 nM T58970 C9A3KO 122193410 IC50 = 2000 nM T58970 CM1JW3 122604219 IC50 < 0.3 nM T58970 C2UO3Y 122604256 IC50 = 0.3 nM T58970 C65QNK 122604287 IC50 < 0.3 nM T58970 C2HZB8 122604308 IC50 < 0.3 nM T58970 CGT97F 122604354 IC50 < 0.3 nM T58970 CW0QT8 126480560 IC50 < 0.3 nM T58970 CS8C7J 126480561 IC50 < 1.13 nM T58970 CCIQ37 126480562 IC50 = 2.5 nM T58970 CGY2L4 126480563 IC50 < 0.3 nM T58970 CJM59E 126480564 IC50 < 0.3 nM T58970 CO9CY8 126480565 IC50 = 23 nM T58970 CHQ71G 126480566 IC50 = 2.8 nM T58970 COF75Z 126970673 IC50 = 600 nM T58970 C0HN2Y 127030123 IC50 = 5250 nM T58970 C7S9GI 127030124 IC50 > 100000 nM T58970 CHGN68 127030424 IC50 = 2340 nM T58970 CRV62L 127030425 IC50 > 100000 nM T58970 CF7JT8 127030426 IC50 > 100000 nM T58970 C5YCU2 127030427 IC50 > 100000 nM T58970 C0GES2 127031075 IC50 > 100000 nM T58970 CFJ32Y 127031076 IC50 > 100000 nM T58970 CC8V4J 127031368 IC50 > 100000 nM T58970 C78GYH 127031383 IC50 > 100000 nM T58970 C5WA9Z 127031384 IC50 > 100000 nM T58970 CD7LN1 127031385 IC50 = 1420 nM T58970 CI0VX4 127031386 IC50 > 100000 nM T58970 CO89TC 127031387 IC50 = 1440 nM T58970 CAM4S5 127031675 IC50 > 100000 nM T58970 C4QD0M 127031676 IC50 = 23240 nM T58970 C0LTC3 127031677 IC50 > 100000 nM T58970 CO1G2K 127032542 IC50 > 31600 nM T58970 C12IOL 127033165 IC50 > 100000 nM T58970 C5RO0L 127033758 IC50 > 100000 nM T58970 CD04YX 127034308 IC50 > 31600 nM T58970 CQ1V6G 127045826 IC50 = 7.9 nM T58970 C6KL7C 127045928 IC50 = 12.6 nM T58970 CHK16Q 127045929 IC50 = 53.1 nM T58970 CD13VL 127045930 IC50 = 468.6 nM T58970 CDOK30 127045931 IC50 = 25.8 nM T58970 CF4XM2 127045932 IC50 = 58.9 nM T58970 CC9FG2 127045933 IC50 = 7 nM T58970 CBQ2N5 127046246 IC50 = 219 nM T58970 CLM41O 127046585 IC50 = 9.5 nM T58970 CWRM04 127046871 IC50 = 61.1 nM T58970 CEA32D 127047009 IC50 = 139.5 nM T58970 CO6Q4N 127047015 IC50 = 16.7 nM T58970 CTCR73 127047016 IC50 = 31.3 nM T58970 CA7Z9H 127047017 IC50 = 153.7 nM T58970 C6AVN3 127047018 IC50 = 11.9 nM T58970 CLG53I 127047019 IC50 = 24.1 nM T58970 C2HO7X 127047025 IC50 = 276.4 nM T58970 C0CW2H 127047026 IC50 = 297 nM T58970 CK49NV 127047027 IC50 = 17.9 nM T58970 C3WGY8 127047160 IC50 = 19.4 nM T58970 C4JP8F 127047161 IC50 = 424.6 nM T58970 CZ3NX1 127047176 IC50 = 15.6 nM T58970 CUI42E 127047178 IC50 = 109.5 nM T58970 CKQU80 127047563 IC50 = 63.3 nM T58970 CG89KZ 127047589 IC50 = 9.3 nM T58970 CLO6T3 127047590 IC50 = 22.5 nM T58970 CY3J0C 127047591 IC50 = 16.7 nM T58970 C5KVU1 127047600 IC50 = 632 nM T58970 CD6X7F 127047723 IC50 = 225.8 nM T58970 CKQ9P4 127047724 IC50 = 13.2 nM T58970 CO6DK5 127047745 IC50 = 50.6 nM T58970 CQKW20 127048111 IC50 > 2000 nM T58970 CE17QJ 129053010 IC50 = 420 nM T58970 CS27PK 129053060 IC50 = 2.5 nM T58970 C6GP3F 129053136 IC50 = 4.2 nM T58970 CJ4NM9 129053223 IC50 = 11 nM T58970 C89SUW 129053289 IC50 = 4 nM T58970 CV7IZ4 129053305 IC50 = 4.3 nM T58970 C1U6LF 129053491 IC50 = 3 nM T58970 CBI0J3 129077199 IC50 = 4.1 nM T58970 CF37PW 129077224 IC50 = 24 nM T58970 CE8CZ5 129077298 IC50 = 40 nM T58970 CGD6H8 129077301 IC50 = 68 nM T58970 C8QA1C 129077798 IC50 = 7.9 nM T58970 C4ZKE2 129077836 IC50 = 21 nM T58970 C6OQ0F 129077890 IC50 = 26 nM T58970 CUD5M2 129077995 IC50 = 2.1 nM T58970 CBSW14 129116690 IC50 < 0.3 nM T58970 C2ZO8R 129116708 IC50 < 0.3 nM T58970 CS6OA8 129116809 IC50 = 0.83 nM T58970 CV98PG 129136448 IC50 < 0.3 nM T58970 C2LWZ1 129318964 IC50 > 10000 nM T58970 C8ARK0 131801160 IC50 = 1090 nM T58970 C0AV5D 131801161 IC50 = 90.3 nM T58970 CB3C0Z 132819859 IC50 = 277 nM T58970 CK6Z5F 132819860 IC50 > 10000 nM T58970 CR3C9O 132819862 IC50 = 7890 nM T58970 CAG60V 132819865 IC50 = 3140 nM T58970 CE4Z3X 132819866 IC50 = 242 nM T58970 CITU18 134129122 IC50 = 76000 nM T58970 C3TW9Y 134130036 IC50 = 4620 nM T58970 CTDB31 134130124 IC50 > 10000 nM T58970 C5N0CA 134130303 IC50 = 225 nM T58970 C4S7VK 134130361 IC50 = 1670 nM T58970 C2IB7F 134130412 IC50 = 736 nM T58970 CH7A9R 134130612 IC50 = 5600 nM T58970 CEH49U 134130924 IC50 = 361 nM T58970 COL93E 134131237 IC50 = 9230 nM T58970 CZ31WJ 134132433 IC50 = 24.3 nM T58970 C3L0ZC 134140633 IC50 = 118.2 nM T58970 C2AN7T 134611886 IC50 > 100000 nM T58970 CS4OW8 135400873 Ki = 2000 nM T58970 CXQ03H 135413555 IC50 = 6 nM T58970 CW0P1Q 135433657 IC50 = 89 nM T58970 CI1JQ3 135449325 Ki = 86 nM T58970 C8GZ2B 135449326 Ki = 2 nM T58970 C3F9CW 135453331 Ki = 230 nM T58970 C4Q5CE 135453643 Ki < 1000 nM T58970 CO6I2L 135523935 Ki = 580 nM T58970 C1Q2AL 135523936 Ki = 870 nM T58970 C2PQT5 135523937 Ki > 10000 nM T58970 CP2B4U 135523938 Ki = 440 nM T58970 C0GMF7 135523939 Ki = 490 nM T58970 CSI4D2 135523940 Ki = 330 nM T58970 COM67B 135523941 Ki = 100 nM T58970 CX56SF 135523946 Ki = 35 nM T58970 CWU14F 135523947 Ki = 510 nM T58970 CX5LG4 135523948 Ki = 2300 nM T58970 CNY53K 135523949 Ki = 63 nM T58970 C1HUP6 135523950 Ki = 44 nM T58970 CA7HF8 135523951 Ki = 24 nM T58970 CT08OB 135523952 Ki = 7 nM T58970 C28SDI 135523953 Ki = 150 nM T58970 CJ08EW 135523954 Ki = 200 nM T58970 CZ87OT 135523955 Ki = 430 nM T58970 C0ZL3Y 135523956 Ki = 2000 nM T58970 C5Q0GA 135523957 Ki = 40 nM T58970 CF2G9Y 135523958 Ki = 510 nM T58970 CGHE70 135523959 Ki = 170 nM T58970 CWZ6R0 135523960 Ki = 660 nM T58970 CIHM29 135523961 Ki > 5000 nM T58970 CHW83U 135523962 Ki = 4000 nM T58970 CD1G6A 135523963 Ki = 14 nM T58970 CA41BZ 135523964 Ki = 240 nM T58970 C4JCM5 135523965 Ki = 22 nM T58970 C51XUS 135523966 Ki = 6 nM T58970 CTJ48K 135524085 IC50 = 2600 nM T58970 CUT1W7 135524168 IC50 = 1100 nM T58970 CYD9P2 135529466 Ki = 160 nM T58970 CRJ45X 135589980 IC50 > 50000 nM T58970 CFAD48 135611170 Ki = 220 nM T58970 CDOJ10 135882424 IC50 = 47000 nM T58970 CYDM01 135891431 IC50 > 10000 nM T58970 CHA4N2 136013680 IC50 > 10 nM T58970 C26ESH 136060555 IC50 > 50000 nM T58970 C3I2CY 136065819 IC50 > 100000 nM T58970 CAW0E4 136065882 IC50 = 702 nM T58970 CUH08T 136094929 IC50 = 12400 nM T58970 C1YUD0 136219394 IC50 > 10 nM T58970 COG2M5 136242661 Ki = 1160 nM T58970 CM63AX 136245248 Ki = 1000000 nM T58970 CIU8W3 136254389 IC50 > 10 nM T58970 CZTI25 136623676 IC50 = 940 nM T58970 CG67XB 137210065 IC50 = 32.9 nM T58970 C0CV4B 137210066 IC50 = 22.4 nM T58970 C04YDK 137248544 Ki = 3000 nM T58970 CMB78I 137301774 Ki = 19000 nM T58970 C01QHB 137348765 IC50 = 160 nM T58970 C25ERN 137631967 IC50 > 1000 nM T58970 CO19HF 137633457 IC50 = 370 nM T58970 CM2VQ1 137636104 IC50 < 0.3 nM T58970 C06JRX 137637094 IC50 = 574.7 nM T58970 CZAM24 137638642 IC50 = 13 nM T58970 CTI5H6 137641993 IC50 = 0.2 nM T58970 CCO7X8 137643676 IC50 = 1.9 nM T58970 C07BXP 137644714 IC50 < 0.3 nM T58970 CDA2N6 137644922 IC50 = 61 nM T58970 CTDK87 137646412 IC50 = 9.2 nM T58970 C7D1TY 137647232 IC50 < 0.39 nM T58970 CN9A1C 137647463 IC50 = 2.7 nM T58970 C5M9VT 137649141 IC50 < 0.34 nM T58970 C0VRK3 137651050 IC50 = 25 nM T58970 C1DK0P 137651391 IC50 > 1000 nM T58970 CH2JO0 137651415 IC50 = 14 nM T58970 CI46SD 137652179 IC50 = 1.4 nM T58970 CC32NU 137654819 IC50 < 0.31 nM T58970 CV5H3Z 137657932 IC50 = 960.2 nM T58970 C6J5TG 137658266 IC50 < 0.48 nM T58970 C4P2JF 137659314 IC50 = 3.7 nM T58970 CD1P2J 137660437 IC50 = 12300 nM T58970 CAL90E 137660905 IC50 = 700 nM T58970 C3W4RO 138403252 IC50 = 850000 nM T58970 CYZ5E0 143488659 IC50 = 25 nM T58970 C6VB3O 145925651 IC50 >= 5000 nM T58970 C5TS1A 145964021 IC50 = 13 nM T58970 C8QAU0 145965069 IC50 = 291 nM T58970 C3Z6FW 145965114 IC50 = 729 nM T58970 CGY5U6 145967586 IC50 = 5.8 nM T58970 CDNC31 145967951 IC50 > 500 nM T58970 CB13TD 145968084 IC50 = 90 nM T58970 CVE53B 145968293 IC50 = 960 nM T58970 CQJP12 145968722 IC50 = 13 nM T58970 C51ZYU 145968739 IC50 = 15.5 nM T58970 CDWJ18 145969577 IC50 > 1000 nM T58970 CPG2Z1 145969751 IC50 = 115 nM T58970 CD7X3A 145969845 IC50 = 29 nM T58970 CQ5FM4 145970383 IC50 = 9.7 nM T58970 C6VH0C 145970689 IC50 = 1311 nM T58970 CGA71R 145970914 IC50 > 3000 nM T58970 CSJ5I2 145971084 IC50 = 574 nM T58970 CG01BZ 145973754 IC50 = 6 nM T58970 C6X8PU 145975686 IC50 = 5 nM T58970 C28XFL 145977776 IC50 = 114 nM T58970 C2FA4R 145978301 IC50 = 5 nM T58970 C8OV5Y 145986581 IC50 = 119 nM T58970 CNR4I2 145987741 IC50 = 14 nM T58970 C3NUY1 146634275 IC50 = 22.3 nM T58970 C58UFW 146634276 IC50 = 0.8 nM T58970 C47CZG 146634277 IC50 = 5.4 nM T58970 CG5K6V 146634280 IC50 = 25.6 nM T58970 C58ZBS 146634281 IC50 > 1000 nM T58970 CV6S1K 146634282 IC50 = 201 nM T58970 CA3NM7 146634283 IC50 = 633 nM T58970 C5UV0A 146634285 IC50 = 1.1 nM T58970 C09IAM 146634730 IC50 = 38.4 nM T58970 C73IJV 146634731 IC50 = 2.7 nM T58970 C3XSK8 146634732 IC50 = 17.8 nM T58970 CD7T9R 146634733 IC50 = 11.2 nM T58970 CVM9Z0 146634734 IC50 = 2.9 nM T58970 CHIB04 146634736 IC50 = 3.6 nM T58970 C3MR9I 146634737 IC50 = 1.9 nM T58970 CC98HU 146634738 IC50 = 3.5 nM T58970 C6Q3UP 146634739 IC50 = 0.7 nM T58970 C5P8GS 146634740 IC50 = 17.6 nM T58970 CX76AZ 146634741 IC50 = 1.2 nM T58970 CSZQ50 146634742 IC50 = 7.2 nM T58970 C10WET 148308905 IC50 = 1.6 nM T58970 CPD47L 148858814 IC50 = 3.1 nM T58970 C1IP0X 155510958 IC50 = 30.4 nM T58970 C2MD1Q 155513187 IC50 > 10000 nM T58970 CC8FG7 155514156 IC50 = 36.3 nM T58970 C86HPW 155518524 IC50 = 66000 nM T58970 CE8JP2 155518580 IC50 > 1000 nM T58970 CLK3T4 155526028 IC50 > 1000 nM T58970 C86ALC 155528265 IC50 > 3000 nM T58970 CNI60D 155530043 IC50 = 2400 nM T58970 C2XM5B 155534129 IC50 = 0.13 nM T58970 CA8XV9 155535222 IC50 = 93.3 nM T58970 C7WAG2 155535552 IC50 = 19.8 nM T58970 C9L0CN 155537763 IC50 = 56 nM T58970 C73PVJ 155545110 IC50 > 1000 nM T58970 CW7MV3 155545248 IC50 > 1000 nM T58970 CE21BL 155553718 IC50 = 5.6 nM T58970 C2K3QV 155556154 IC50 = 35.6 nM T58970 C0XZ5C 155562528 IC50 = 0.7 nM T58970 CYB5S2 155566604 IC50 < 0.3 nM T58970 C5TAN1 155566828 IC50 > 1000 nM T58970 D00ERW 44444843 Ki > 8750 nM T58970 D00HVA 11624601 Ki = 4700 nM T58970 D01MNK 25125014 IC50 = 3110 nM T58970 D01WAI 135451156 IC50 = 824 nM T58970 D01YWE 25207521 IC50 = 4200 nM T58970 D02XHC 448912 IC50 = 22000 nM T58970 D03DZO 11715767 IC50 > 10000 nM T58970 D04ZWF 53396311 IC50 > 10000 nM T58970 D06HVH 54613583 IC50 > 10000 nM T58970 D07ADX 54764565 IC50 = 6290 nM T58970 D08BMM 6312649 IC50 > 2500 nM T58970 D08HFG 24809764 IC50 > 10000 nM T58970 D08XVZ 24866313 IC50 < 0.3 nM T58970 D09HVH 135566652 IC50 > 10 nM T58970 D09XIL 11396738 IC50 = 12600 nM T58970 D0CM6T 11314340 Ki = 260 nM T58970 D0D6MH 11617559 IC50 > 10000 nM T58970 D0EW9J 10389239 IC50 = 3440 nM T58970 D0F0AX 135413546 IC50 = 9 nM T58970 D0I4NN 14056555 IC50 > 2500 nM T58970 D0J3LR 11634725 Ki < 2 nM T58970 D0ME9B 46868971 IC50 > 10 nM T58970 D0O6OH 71553154 IC50 = 30000 nM T58970 D0Q3KS 9957049 IC50 > 10000 nM T58970 D0Q3NG 11715520 Ki > 8800 nM T58970 D0S7IE 11658882 Ki > 8800 nM T58970 D0T8NU 16757525 IC50 = 846 nM T58970 D0TF0V 3085877 IC50 > 2500 nM T58970 D0UN9O 3385203 IC50 >= 10000 nM T58970 D0YZ7H 9797370 IC50 > 100000 nM T58970 D0ZG4G 11493598 Ki = 310 nM T83143 C8K6AO 16187262 IC50 = 1260 nM T83143 CSV0R5 24791838 IC50 = 3360 nM T83143 CI1QX7 24793028 IC50 = 3160 nM T83143 C4H6VD 24793288 IC50 = 760 nM T83143 C0ZLH5 24793407 IC50 = 600 nM T83143 CSE16O 24793875 IC50 = 4470 nM T83143 C6H2KZ 24817638 IC50 = 100 nM T83143 C2BC6P 24819334 IC50 = 4220 nM T83143 C9QCY0 25281482 IC50 = 1560 nM T83143 CE3PH5 26331136 IC50 = 1020 nM T83143 CBH1P0 42210730 IC50 = 1640 nM T83143 C2L9IY 42287393 IC50 = 1850 nM T83143 CT0NF6 42415086 IC50 = 910 nM T83143 C07FPT 42515059 IC50 = 8090 nM T83143 CUL67Y 45202552 IC50 = 1730 nM T83143 C97WSO 70678458 IC50 = 760 nM T83143 CO9TC3 70678478 IC50 = 6120 nM T83143 C3RL6W 70679275 IC50 = 1250 nM T83143 CC6T5K 70679283 IC50 = 72 nM T83143 C43IWS 71453989 IC50 = 3200 nM T83143 C7AYV5 118540795 Ki = 68 nM T83143 CV3UP6 129909861 IC50 = 270 nM T83143 CS5V9K 134134587 IC50 = 467 nM T83143 C13INT 134134961 IC50 > 10000 nM T83143 C0MKT2 134139392 IC50 = 1840 nM T83143 CWO69F 134153091 IC50 = 3350 nM T83143 C9FB8J 134154850 IC50 = 640 nM T83143 D05ZUX 44207909 Ki >= 1000 nM T83143 D0T2RY 9948320 Ki >= 1000 nM T25307 D02DGU 444795 IC50 = 199.53 nM T25307 D02OZE 2724385 IC50 = 4000 nM T25307 D0G3PI 449171 EC50 = 14000 nM T25307 D0BF4Z 89875987 IC50 = 17 nM T25307 D0D7CH 118622692 IC50 = 1.9 nM T25307 D0T7YE 124126348 EC50 = 30.1 nM T25307 C25CAT 122184111 EC50 = 8.1 nM T25307 CVS15Y 122184115 EC50 = 10 nM T25307 C6R8ES 72721387 EC50 = 97 nM T25307 CCW45Q 72721388 EC50 = 93 nM T25307 CQO6D1 6626 IC50 > 10000 nM T25307 CGH93A 73864 IC50 > 10000 nM T25307 CPF05U 92746 EC50 = 110 nM T25307 C2LPT4 99470 EC50 = 20 nM T25307 CA56RZ 168038 EC50 = 20 nM T25307 C5TJ6B 440711 EC50 = 20 nM T25307 C4TID5 623849 IC50 > 10000 nM T25307 CKO0L6 807146 EC50 = 100 nM T25307 CTW4U7 982780 IC50 = 80 nM T25307 CSHG48 1186353 IC50 > 10000 nM T25307 C86NCM 1188393 EC50 > 10000 nM T25307 CZL36X 1249036 IC50 = 380 nM T25307 CKF5R7 1286153 IC50 = 151900 nM T25307 CDRG30 1302006 IC50 = 4540 nM T25307 C5N3FQ 1353440 IC50 = 140 nM T25307 C0A5IB 1367810 IC50 = 300 nM T25307 C83WZI 1523409 IC50 = 90 nM T25307 CP3H7L 1735453 IC50 = 11640 nM T25307 C3EB4O 2055236 IC50 = 5930 nM T25307 CQ7YP2 2245525 IC50 = 37540 nM T25307 CZ8K4H 2279516 IC50 = 27220 nM T25307 CD06AX 2280700 IC50 = 420 nM T25307 C4ZUK2 2339329 IC50 > 25118.86 nM T25307 CNI31L 3278739 IC50 = 1548.82 nM T25307 CZ6LB3 3351335 IC50 = 18270 nM T25307 CO6LR8 3443633 IC50 = 7.5 nM T25307 CNX58C 3595981 IC50 = 168270 nM T25307 C93VEI 4096741 IC50 = 142210 nM T25307 C5U1QL 4303549 IC50 = 8280 nM T25307 C5I2LS 4428639 IC50 = 200 nM T25307 C3C7KJ 4642411 IC50 = 81 nM T25307 CE3K6R 5057409 IC50 = 81690 nM T25307 C8EZJ5 6036629 IC50 = 46870 nM T25307 C0AWF1 6405443 IC50 = 11140 nM T25307 C42OPB 7517782 EC50 = 3600 nM T25307 CC42LQ 7517788 EC50 > 10000 nM T25307 C1BLW8 7517789 EC50 = 550 nM T25307 CMPR10 7517833 EC50 > 10000 nM T25307 C36CNX 8892653 EC50 = 100 nM T25307 C2ZRB1 9617733 IC50 = 56640 nM T25307 C6F2QA 9935973 EC50 = 100 nM T25307 CXA0N9 10458226 EC50 = 4000 nM T25307 CIB9H5 11439236 IC50 = 150 nM T25307 CTD5G1 13799749 IC50 = 216000 nM T25307 C2SKY8 15944563 IC50 = 14090 nM T25307 C1H8JU 15944574 IC50 = 10 nM T25307 CY97FK 16028122 IC50 = 1470 nM T25307 C5LMJ9 16445174 EC50 = 100 nM T25307 C82YFG 16746312 IC50 = 15700 nM T25307 CF60TV 16746329 IC50 = 2500 nM T25307 C0S8XW 16746343 IC50 > 50000 nM T25307 C7G8OT 16746402 IC50 = 3300 nM T25307 CIB0Y1 16746480 IC50 > 50000 nM T25307 C2NX6V 16830309 EC50 = 2100 nM T25307 C6Q8KB 16837923 IC50 = 5011.87 nM T25307 CTG9Z4 16911249 IC50 = 7943.28 nM T25307 CS79UQ 17613473 IC50 = 6060 nM T25307 C0O6CM 17980288 EC50 > 10000 nM T25307 C0CQR1 18565104 IC50 = 180 nM T25307 C4MQ7E 18565133 EC50 = 120 nM T25307 C2LMW1 18565134 EC50 = 43 nM T25307 C0QKH8 18565138 EC50 = 26 nM T25307 CGS1R9 18565141 IC50 < 15000 nM T25307 C8SOP2 18565142 EC50 = 420 nM T25307 C84GPT 18565143 EC50 = 470 nM T25307 CF43IK 18565194 EC50 = 570 nM T25307 CVGU30 18578056 IC50 = 110 nM T25307 C9MQ8H 18586895 IC50 = 3981.07 nM T25307 C2I0YG 18587009 IC50 = 7943.28 nM T25307 CDRB15 18587012 IC50 = 3981.07 nM T25307 CG6WC3 18587019 IC50 = 6309.57 nM T25307 CAC36Q 18587021 Ki = 398.11 nM T25307 CUN47I 18587054 IC50 = 1258.93 nM T25307 CC3VD4 18587059 IC50 > 25118.86 nM T25307 C4RYO8 19760309 IC50 > 10000 nM T25307 C38JEL 20704150 EC50 = 190 nM T25307 C1FJU8 21824365 IC50 = 14500 nM T25307 C38CHU 24776335 EC50 > 10000 nM T25307 C1BIA8 24906344 IC50 = 1350 nM T25307 CX2Q9M 24906350 IC50 = 5150 nM T25307 CF1S8P 25132150 IC50 > 20000 nM T25307 CNG1Z5 25132504 IC50 = 9000 nM T25307 CB56QH 25132505 IC50 > 20000 nM T25307 CS1EJ7 25234324 EC50 = 360 nM T25307 CP6I8T 27545839 EC50 > 10000 nM T25307 CGMR40 27548891 EC50 = 1700 nM T25307 CAQ1L7 27557585 EC50 > 10000 nM T25307 C8KAR1 30171711 IC50 = 1030 nM T25307 C35PLM 30171813 IC50 = 1390 nM T25307 C3V4WB 38023871 IC50 = 19000 nM T25307 CZ34LM 41145772 IC50 = 1258.93 nM T25307 CO1NQ0 41145803 IC50 = 15.85 nM T25307 CGY80Q 44409326 IC50 = 883 nM T25307 CV8TS3 45573446 EC50 = 7400 nM T25307 C1UE6W 45573449 EC50 = 6800 nM T25307 CGT01Z 45573451 EC50 > 10000 nM T25307 C9ZWM8 46866594 IC50 = 3900 nM T25307 CMR49F 46885348 IC50 > 20000 nM T25307 C18JYQ 46885349 IC50 = 5800 nM T25307 C4TLX3 46885390 IC50 = 16800 nM T25307 CSP3D8 46885467 IC50 = 9200 nM T25307 C8WM2R 46885468 IC50 = 11900 nM T25307 CP3O2L 46885469 IC50 > 20000 nM T25307 CG6JE7 46885508 IC50 = 10400 nM T25307 CX2U0L 46886033 IC50 > 20000 nM T25307 C6J5RT 46886034 IC50 = 4700 nM T25307 CV5IN9 46943306 IC50 = 114 nM T25307 CY0JK1 46943315 IC50 = 30000 nM T25307 CWO20S 46943319 IC50 = 3300 nM T25307 CN06IL 46943323 IC50 = 57 nM T25307 CJLT51 46943332 IC50 = 29000 nM T25307 CPVL46 46943335 IC50 = 4700 nM T25307 CYK9B5 46943340 IC50 > 1000 nM T25307 CPB51M 46943341 IC50 > 50000 nM T25307 CMQ94N 46943368 IC50 = 22500 nM T25307 C9DAR7 46943373 IC50 = 6600 nM T25307 C8JYP1 46943390 IC50 = 24400 nM T25307 CM9TJ3 46943394 IC50 > 1000 nM T25307 C8P6MQ 46943400 IC50 = 12800 nM T25307 CN8C4X 46943404 IC50 = 4000 nM T25307 C40VNC 51035446 IC50 = 90 nM T25307 C4F9RZ 51035449 Ki = 105 nM T25307 C2GN8U 51344321 IC50 = 3990 nM T25307 CMN53E 51344322 IC50 = 12770 nM T25307 C14MKP 51344334 IC50 = 93850 nM T25307 CT0F9J 52100402 IC50 = 200 nM T25307 CM7BY6 53385590 IC50 = 51 nM T25307 CC9J5N 53390693 IC50 > 1000 nM T25307 C2P5HX 54582225 IC50 = 9200 nM T25307 CQ02IF 54582227 IC50 > 10000 nM T25307 CS9O7F 54582228 IC50 = 1100 nM T25307 CPF9X2 54587076 IC50 = 5700 nM T25307 CFO23H 56837193 EC50 = 8 nM T25307 CF6I8J 56847994 IC50 = 10 nM T25307 CL9T0Q 56848043 IC50 = 7943.28 nM T25307 CYZG78 56848095 IC50 = 39.81 nM T25307 CAI2T0 56848145 IC50 = 31.62 nM T25307 C4UK1P 57521299 IC50 = 7.943 nM T25307 C7A0YE 57521310 IC50 = 6 nM T25307 CWF63S 59054468 IC50 = 10 nM T25307 CI24SQ 59054496 IC50 = 15.85 nM T25307 CH3I4A 60142604 IC50 = 39.81 nM T25307 C9ETS7 60142605 IC50 = 398.11 nM T25307 CP2R5C 60142606 IC50 = 12.59 nM T25307 CZP7J9 60142607 IC50 = 630.96 nM T25307 CVM95C 60142739 IC50 = 15.85 nM T25307 CB91KH 60142741 IC50 = 10 nM T25307 CN4V9K 60142742 IC50 = 19.95 nM T25307 C0P3BH 60142867 IC50 = 19.95 nM T25307 C0AF3D 60142996 IC50 = 199.53 nM T25307 CB07HN 60142998 IC50 = 12.59 nM T25307 CZE4U3 60162553 EC50 = 11 nM T25307 C6OBI4 60162810 EC50 = 68 nM T25307 C7P2TS 60243771 IC50 = 170 nM T25307 COQR02 66554786 EC50 < 500 nM T25307 CLO85B 66562432 EC50 < 500 nM T25307 CDF9R6 66562538 EC50 < 500 nM T25307 C2JNE3 67418549 EC50 < 500 nM T25307 CONJ97 68159303 IC50 = 2 nM T25307 CI8P2A 68159594 IC50 = 958 nM T25307 CI8U4Z 68233447 EC50 < 500 nM T25307 CDM9Q3 68276046 IC50 = 12.59 nM T25307 C1FGP2 68276052 IC50 = 12.59 nM T25307 CJ8HV4 68276072 IC50 = 110 nM T25307 C3XRP1 68277108 IC50 = 6.31 nM T25307 CE1DV5 68277124 IC50 = 10 nM T25307 C0TIW1 68277128 IC50 = 7.943 nM T25307 CP6N4Y 68278907 IC50 = 3 nM T25307 C1URW8 68278937 IC50 = 586 nM T25307 CP8BU3 68279056 EC50 < 50 nM T25307 CGD5T0 68279070 EC50 < 50 nM T25307 C7T8RU 68279071 IC50 = 6 nM T25307 C3EST0 69282351 IC50 < 15000 nM T25307 CJ0I1V 71082496 IC50 = 13000 nM T25307 C0GW6I 71127425 EC50 = 2300 nM T25307 C6Z3NE 71127467 EC50 = 71 nM T25307 C6VK1N 71127470 EC50 = 320 nM T25307 C8E1DZ 71135801 EC50 = 44 nM T25307 CVY3G8 71247311 IC50 = 17 nM T25307 CC6P1F 71247312 IC50 = 33 nM T25307 CQK0X1 71247410 IC50 = 1 nM T25307 CMD9H6 71251176 IC50 = 1 nM T25307 CGD2C7 71283712 IC50 = 100 nM T25307 CL6T1F 71283714 IC50 = 7.943 nM T25307 CBG9Q4 71283798 IC50 = 5.012 nM T25307 CEO15M 71283813 IC50 = 6.31 nM T25307 C0S5QO 71283824 EC50 = 1 nM T25307 CCS2X9 71283851 IC50 = 6.31 nM T25307 C3BS8U 71283919 IC50 = 6.31 nM T25307 C9D0PC 71283954 IC50 = 3.981 nM T25307 C2IS3B 71283966 IC50 = 7.943 nM T25307 CTQ49I 71283975 IC50 > 25118.86 nM T25307 CO0B2L 71285679 IC50 = 10 nM T25307 C9E8VD 71285767 IC50 = 31.62 nM T25307 CRHQ21 71285777 IC50 = 3.162 nM T25307 CZY93F 71285783 IC50 = 5.012 nM T25307 CG3U8E 71285798 IC50 = 5.012 nM T25307 CY9Q5G 71285802 IC50 = 6.31 nM T25307 CSY0B9 71285807 IC50 = 63.1 nM T25307 C98PDI 71285817 IC50 = 5.012 nM T25307 C61MTB 71285820 IC50 = 15.85 nM T25307 CCJ5K1 71285825 IC50 = 7943.28 nM T25307 CZ8I2P 71285829 EC50 = 1 nM T25307 CR2KO6 71285842 IC50 = 398.11 nM T25307 C7PLS6 71285927 IC50 = 112 nM T25307 C7D8WL 71285944 IC50 = 3.981 nM T25307 CBQ7U5 71286169 IC50 = 31.62 nM T25307 CA83DQ 71286208 IC50 = 10 nM T25307 CIL4M0 71286223 EC50 = 1 nM T25307 C4UH5M 71289906 IC50 = 1000 nM T25307 C1MLW3 71289939 IC50 = 6.31 nM T25307 CJNU36 71289978 IC50 = 3.981 nM T25307 CFGP17 71289981 IC50 = 10 nM T25307 CP5GL9 71470549 Ki = 1000 nM T25307 CSA28U 71470550 IC50 = 430 nM T25307 C5FN9O 71470724 IC50 = 70 nM T25307 CS23YJ 71492470 IC50 = 1 nM T25307 C8P0WC 71492999 IC50 = 1 nM T25307 CL5P3W 71494750 IC50 = 1 nM T25307 C2YAK1 71508397 IC50 = 5.9 nM T25307 CD9FE7 71538152 IC50 = 1.6 nM T25307 CG7O8L 71540054 IC50 = 106 nM T25307 C4Q3WF 71540059 IC50 > 1000 nM T25307 CZQ89H 71540280 IC50 > 1000 nM T25307 CO6U2Y 71540281 IC50 > 1000 nM T25307 CTJK70 71540282 IC50 > 1000 nM T25307 CVU0W7 71540284 IC50 > 1000 nM T25307 CK50WA 71540632 IC50 = 800 nM T25307 C1UQF6 71540740 IC50 = 800 nM T25307 CZO9K0 71540741 IC50 = 1000 nM T25307 CQ53UO 71540742 IC50 = 800 nM T25307 C2T4IL 71540858 IC50 = 1700 nM T25307 CDJV35 71540859 IC50 = 1000 nM T25307 C9JBU5 71543524 IC50 < 16 nM T25307 C1UIH6 71543682 EC50 < 16 nM T25307 CK1FA9 71557114 EC50 < 500 nM T25307 CJHD64 71557116 EC50 < 500 nM T25307 C71EWG 71582623 EC50 = 16 nM T25307 CS83WA 71612299 IC50 = 18 nM T25307 C71SQK 71612302 EC50 = 4 nM T25307 C0H7LK 71612419 EC50 = 9 nM T25307 CXK08C 71612420 EC50 = 3 nM T25307 CNP23X 71612421 EC50 = 11 nM T25307 CA8IC6 71612422 EC50 = 6 nM T25307 CFCK26 71612423 IC50 = 7 nM T25307 C1DR8E 71622396 EC50 = 21 nM T25307 C8CZX6 71622397 IC50 = 31 nM T25307 C3WX1L 71622670 EC50 = 200 nM T25307 CE3CU6 71622672 EC50 = 2700 nM T25307 C6YKL7 71622674 IC50 = 120 nM T25307 C2QOV7 71719136 IC50 > 1000 nM T25307 C6BGN1 71719745 IC50 > 1000 nM T25307 C65ZCF 71811962 EC50 < 10000 nM T25307 C1XJ0R 72165233 EC50 < 50 nM T25307 CW5U4Q 72189290 EC50 = 32 nM T25307 CGW3N9 72193937 EC50 = 20 nM T25307 CLZ0T9 72194571 EC50 < 10000 nM T25307 CJ3I8D 72194692 EC50 < 32 nM T25307 C14KPM 72548240 EC50 = 10000 nM T25307 CWH6T3 72548703 EC50 = 2.8 nM T25307 CIV80W 72548704 EC50 = 1 nM T25307 CX0H3D 72548705 IC50 = 12 nM T25307 CZ0P6M 72548955 IC50 = 1.8 nM T25307 CJGR93 72548957 IC50 = 2.6 nM T25307 C1R2CH 72549410 IC50 = 28 nM T25307 CFLV24 72700652 EC50 < 10000 nM T25307 CDXN75 72706017 EC50 = 450 nM T25307 CM5YU9 72720561 IC50 = 10000 nM T25307 C32FIQ 72720562 EC50 = 450 nM T25307 CQ0UK6 72720563 EC50 = 530 nM T25307 CSM3D2 72720564 EC50 = 210 nM T25307 CC8YU6 72720884 EC50 = 200 nM T25307 CXY34A 72720885 IC50 = 100 nM T25307 CJ3W7N 72720886 EC50 = 160 nM T25307 C5WY8U 72720887 IC50 = 2100 nM T25307 C16ALF 72720888 EC50 = 210 nM T25307 C3R9EH 72720985 EC50 = 330 nM T25307 CU9F0Q 72720988 IC50 = 1340 nM T25307 CE73WQ 72721804 IC50 = 89 nM T25307 C3QZT8 72721991 IC50 = 10900 nM T25307 CHE7J8 72721992 IC50 = 6200 nM T25307 CPB51D 72721993 IC50 = 9300 nM T25307 CX8TF5 72722090 IC50 = 1000 nM T25307 C2D7HA 72722091 EC50 = 140 nM T25307 CT6SF0 72722092 IC50 = 200 nM T25307 CC1R6Q 72722093 IC50 = 3600 nM T25307 CJ3CP5 72722095 IC50 = 4800 nM T25307 C61ZIQ 72722443 IC50 = 3000 nM T25307 C3OHQ9 72722444 EC50 > 10000 nM T25307 C65YOG 72722445 EC50 > 10000 nM T25307 CV5D9O 72722446 EC50 > 10000 nM T25307 C9OW7Q 72722447 EC50 = 4000 nM T25307 C1B2WF 72722806 IC50 = 520 nM T25307 CMZ85K 72722807 EC50 = 61 nM T25307 CLT37A 72722808 EC50 = 20 nM T25307 C2BQO3 72722945 EC50 = 19 nM T25307 C4YIT3 72722946 IC50 = 748 nM T25307 CR9VF2 72722948 IC50 = 5000 nM T25307 CNA8Q9 72722949 IC50 = 520 nM T25307 C3HN1C 72722950 EC50 = 1000 nM T25307 CJZH06 72724684 EC50 = 8000 nM T25307 CHR6M9 72724685 EC50 = 9000 nM T25307 CP82IF 72724686 EC50 > 10000 nM T25307 CCK2J7 72724687 EC50 > 10000 nM T25307 CD6A0R 72724688 IC50 = 9000 nM T25307 C29IJM 72724689 IC50 = 329 nM T25307 CLP28Y 72724833 EC50 = 4000 nM T25307 C7QL3U 72943563 IC50 = 1 nM T25307 C6LP9I 73293431 IC50 = 4 nM T25307 C30CNG 73293433 IC50 = 76 nM T25307 C6F8BJ 73293971 IC50 = 300 nM T25307 C6QZE9 73294166 IC50 = 3766 nM T25307 CFY87N 73333084 IC50 > 25118.86 nM T25307 C9YOG8 73333085 IC50 = 10000 nM T25307 CT3BJ6 73333086 IC50 = 5011.87 nM T25307 CR7SM9 73333087 IC50 = 1584.89 nM T25307 C6ZSW8 73333186 IC50 > 25118.86 nM T25307 C87LPH 73333187 IC50 = 1258.93 nM T25307 C0M6NI 73333188 IC50 = 12589.25 nM T25307 CD85GT 73333189 IC50 > 25118.86 nM T25307 C4QAJ9 73333190 IC50 = 1584.89 nM T25307 CHW6E1 73333286 IC50 = 1995.26 nM T25307 C7V0EJ 73333287 IC50 = 3981.07 nM T25307 C7YDF1 73333288 IC50 = 794.33 nM T25307 C70FAX 73333289 IC50 = 6309.57 nM T25307 CW63YF 73333290 IC50 = 10000 nM T25307 CXS2G0 73333389 IC50 = 5011.87 nM T25307 C2F0BZ 73333390 IC50 = 1995.26 nM T25307 CJ3RZ8 73333391 IC50 = 10000 nM T25307 CYE54L 73333392 IC50 = 2511.89 nM T25307 CO04CL 73333393 IC50 = 25.12 nM T25307 CW57BH 73333484 IC50 = 39.81 nM T25307 C9ZTS6 73333485 IC50 = 12.59 nM T25307 CN5LB2 73333486 IC50 = 794.33 nM T25307 C49XUM 73333487 IC50 = 10 nM T25307 C9VK5E 73333488 IC50 = 12.59 nM T25307 C5J3IS 73333576 IC50 = 19.95 nM T25307 CG1JV4 73333577 IC50 = 25.12 nM T25307 C18NTY 73334657 IC50 > 25118.86 nM T25307 CX9YF7 73671284 IC50 = 5 nM T25307 CMD9H4 73671285 EC50 = 6 nM T25307 C6ZD8B 74220546 IC50 = 85 nM T25307 C3ZYM1 74220611 IC50 = 57 nM T25307 C8Q1AL 74220947 IC50 = 6.6 nM T25307 CJ62FH 74221008 IC50 = 120 nM T25307 C1XF8G 74221009 IC50 = 45 nM T25307 CH97FV 74221196 IC50 = 350 nM T25307 CTN1Z5 74221202 IC50 = 3.9 nM T25307 COQD42 74221204 IC50 = 2.5 nM T25307 CAFB63 74221267 IC50 = 62 nM T25307 C05BXA 74221465 IC50 = 140 nM T25307 C5ZF8B 74221745 EC50 = 14 nM T25307 CAL17U 74221833 EC50 = 62 nM T25307 CZ71XR 74221837 EC50 = 56 nM T25307 C06FXI 74221839 EC50 = 120 nM T25307 CN3V2E 74221923 EC50 = 660 nM T25307 CNL14D 74222010 EC50 = 1000 nM T25307 CBN09Z 74222048 IC50 = 140 nM T25307 CQB9S3 74222221 IC50 = 13 nM T25307 CB08IU 74222308 IC50 = 25 nM T25307 CF79OD 74222808 IC50 = 600 nM T25307 C6MY5O 74222810 IC50 = 50 nM T25307 C3BIV1 74222902 IC50 > 6000 nM T25307 C6UWO5 74762670 EC50 = 6 nM T25307 C1NCZ2 76282979 IC50 = 160 nM T25307 CJXG25 76284182 EC50 = 19 nM T25307 CT2BF9 76310256 IC50 = 20 nM T25307 CXS19B 76310263 EC50 = 25 nM T25307 CRQD23 76313943 IC50 = 79 nM T25307 C0Y2CK 76313948 IC50 = 6 nM T25307 C5PT4U 76314451 IC50 = 4500 nM T25307 C0GM1A 76317483 IC50 = 3 nM T25307 C1W4CT 76317484 IC50 = 8 nM T25307 C93XZH 76321222 IC50 = 13 nM T25307 C1YB7G 76321223 IC50 = 40 nM T25307 CWO31G 76324829 IC50 = 1259 nM T25307 CUS20L 76324830 IC50 = 16 nM T25307 CZX50K 76324831 IC50 = 4 nM T25307 C6AT4N 76328385 IC50 = 4 nM T25307 CDZ28I 76328386 IC50 = 6 nM T25307 CXE9Z6 76332062 IC50 = 6 nM T25307 CGZ72M 76332063 IC50 = 6 nM T25307 C4ANV6 76332069 IC50 = 25 nM T25307 C76XVG 76332070 EC50 = 20 nM T25307 C84JBH 76335675 IC50 = 100 nM T25307 CMW6O1 77620538 IC50 = 130 nM T25307 C7ZMD9 78319220 IC50 = 690 nM T25307 C37RIM 78324933 IC50 = 7.2 nM T25307 C4P0KM 82494716 IC50 > 500000 nM T25307 CGTP63 86277915 IC50 = 180 nM T25307 CB7H4C 86288875 IC50 = 40 nM T25307 CEI4V3 86288876 IC50 = 20 nM T25307 C4SA8H 86302482 IC50 = 31 nM T25307 C6HN8M 86346644 EC50 = 69 nM T25307 CBI06J 86346645 EC50 = 57 nM T25307 C72JVE 86566371 IC50 = 4.3 nM T25307 C68WSB 86686467 EC50 = 190 nM T25307 C5VCM4 86690644 EC50 = 30 nM T25307 CGFW70 86690646 EC50 = 13 nM T25307 C0MFA1 86690653 EC50 = 29 nM T25307 CV2L9A 86715668 IC50 = 46 nM T25307 C0FGJ3 86716106 IC50 = 2700 nM T25307 CK9ET8 86716113 IC50 = 110 nM T25307 C4R0OM 86716129 IC50 = 11 nM T25307 C32HDA 86716130 IC50 = 110 nM T25307 C9P0NG 86716147 IC50 = 190 nM T25307 CK98IP 86721886 EC50 = 85 nM T25307 CWK62O 86721898 IC50 = 14 nM T25307 CJ30HZ 86729718 IC50 > 10000 nM T25307 C0QA4G 86729719 IC50 = 190 nM T25307 C2EGM9 86729728 IC50 = 4.8 nM T25307 CQEI47 86729729 IC50 = 140 nM T25307 C4G0ZQ 86729731 IC50 = 15 nM T25307 CR09AC 86729759 IC50 = 57 nM T25307 CJ5D4S 87055114 IC50 = 3.2 nM T25307 CNL0R1 87074581 IC50 = 13 nM T25307 CXO3F6 87085264 IC50 > 40000 nM T25307 C5DW8X 87085361 IC50 > 40000 nM T25307 C7UAI9 88920218 IC50 = 9.4 nM T25307 C43BOV 88920230 IC50 = 10 nM T25307 CUEP93 88920235 IC50 = 131 nM T25307 C0DEZ7 88920270 IC50 = 84 nM T25307 CUP6M0 88924610 IC50 = 31.62 nM T25307 C9TIP6 88924659 IC50 = 398.11 nM T25307 CIW83N 88925021 IC50 = 31.62 nM T25307 C3JH1S 89555559 EC50 < 500 nM T25307 C08ZGH 89607373 EC50 = 40 nM T25307 CI7RX2 89659210 IC50 = 22 nM T25307 CM5LZ4 89659214 EC50 = 10 nM T25307 CI4J1Q 89659216 EC50 = 33 nM T25307 C4F0IR 89659219 IC50 = 220 nM T25307 CR6O7P 89659229 IC50 = 6 nM T25307 C3T9ML 89659363 EC50 = 310 nM T25307 CLSM47 89659364 IC50 = 76 nM T25307 CKB0T4 89659366 EC50 = 4900 nM T25307 CKJE05 89659367 EC50 = 5100 nM T25307 C49MFX 89659368 EC50 = 100 nM T25307 CR49XI 89659369 EC50 = 94 nM T25307 CH51EP 89659380 EC50 = 190 nM T25307 C9WF4L 89659406 EC50 = 160 nM T25307 C31CTH 89659412 EC50 = 70 nM T25307 CA7EC6 89659414 EC50 = 680 nM T25307 C5MOV2 89659415 EC50 = 37 nM T25307 C3PZ1L 89659420 IC50 = 120 nM T25307 CIU47V 89659425 EC50 = 14 nM T25307 CN4PK8 89659438 EC50 = 100 nM T25307 CPM5H8 89659439 EC50 = 6500 nM T25307 C5N0CG 89659441 EC50 = 26 nM T25307 C7RC2B 89659443 EC50 = 310 nM T25307 CCVM78 89659446 EC50 = 47 nM T25307 CW93RI 89659447 EC50 = 41 nM T25307 CV1TN0 89659448 EC50 = 920 nM T25307 C8E2IT 89659450 EC50 = 300 nM T25307 CRO12Y 89659457 EC50 = 63 nM T25307 C4NW8Q 89659463 IC50 = 280 nM T25307 C5L8JQ 89659469 IC50 = 29 nM T25307 CCMG38 89665022 EC50 = 1600 nM T25307 C63RFD 89665043 IC50 = 3600 nM T25307 C8JDQ3 89665048 IC50 = 1500 nM T25307 CLW3O5 89665055 EC50 = 32 nM T25307 CBLJ12 89665057 EC50 = 130 nM T25307 CLUD20 89665061 IC50 = 610 nM T25307 C5HA1W 89665064 IC50 = 2000 nM T25307 C8O9MD 89700756 EC50 = 4900 nM T25307 C5Y1AC 89700815 IC50 = 5400 nM T25307 COP6G8 89700962 EC50 = 23000 nM T25307 CUL15T 89701026 EC50 = 150 nM T25307 CU39CG 89701066 EC50 = 700 nM T25307 CWJ96D 89701093 EC50 = 70 nM T25307 CQ1YI8 89701097 EC50 = 7 nM T25307 C5XBR8 89701100 EC50 = 210 nM T25307 CU1NX6 89701127 EC50 = 860 nM T25307 C86OIZ 89701132 EC50 = 74 nM T25307 CU92ZH 89701145 EC50 = 210 nM T25307 CZGV58 89701201 EC50 = 160 nM T25307 C2VR0P 89701217 IC50 = 24 nM T25307 C3D1UA 90021191 EC50 = 246 nM T25307 C75HQK 90021432 IC50 = 8700 nM T25307 CYZ91N 90030617 IC50 = 1900 nM T25307 CLUP15 90058650 IC50 = 51 nM T25307 CFZL74 90058651 IC50 = 53 nM T25307 CKW01X 90058801 IC50 = 1188 nM T25307 C6H8OJ 90077929 IC50 = 1930 nM T25307 C9K8ID 90077930 IC50 = 2090 nM T25307 CUR34D 90077933 EC50 = 772 nM T25307 CV5Y0H 90077960 IC50 = 50 nM T25307 CNFI27 90077964 EC50 = 58 nM T25307 C6NU9M 90077969 IC50 = 54 nM T25307 CHS95L 90077977 IC50 = 4220 nM T25307 C4CXV6 90077986 IC50 = 1290 nM T25307 C0SCG8 90077990 IC50 = 8100 nM T25307 CE5MU8 90078019 IC50 = 750 nM T25307 C1ZWE8 90078021 IC50 = 1600 nM T25307 CNA5I1 90078028 EC50 < 100 nM T25307 C1VCI2 90078039 IC50 = 2120 nM T25307 CZ24OE 90078100 IC50 = 13000 nM T25307 C41RLB 90078148 EC50 = 717 nM T25307 C0IM3W 90078164 IC50 = 1900 nM T25307 CDZK23 90078179 EC50 = 58 nM T25307 C3OAB9 90078236 IC50 = 3 nM T25307 CQOT46 90078238 IC50 = 1500 nM T25307 CL39VF 90078239 EC50 = 350 nM T25307 C0VFM4 90078240 IC50 = 370 nM T25307 CW5DA3 90088402 IC50 < 15000 nM T25307 CA13SY 90100965 IC50 = 220 nM T25307 CH7U0J 90101666 IC50 = 1000 nM T25307 C18EVT 90130762 EC50 = 98 nM T25307 CGN3K4 90130771 EC50 = 140 nM T25307 CNG7W1 90130850 EC50 = 14000 nM T25307 CQ8JS0 90200433 IC50 = 420 nM T25307 C81URO 90200493 IC50 = 6 nM T25307 C7E5RV 90200534 EC50 = 7 nM T25307 CG83AZ 90200576 IC50 = 440 nM T25307 C81NKB 90200607 IC50 = 93 nM T25307 CTC2K3 90200670 IC50 = 170 nM T25307 CNB93D 90200688 EC50 = 21 nM T25307 C4FX5B 90200758 IC50 = 34 nM T25307 CRM8T6 90200813 IC50 = 510 nM T25307 CJ50LO 90200830 IC50 = 21 nM T25307 CH8S0T 90200856 IC50 = 51 nM T25307 CH4SY0 90200966 IC50 = 61 nM T25307 CZ5WI9 90201077 IC50 = 70 nM T25307 C70HBD 90201096 IC50 = 370 nM T25307 CK59VM 90201157 IC50 = 11 nM T25307 C5GH2Z 90201160 EC50 = 60 nM T25307 C0K2JM 90201176 IC50 = 5600 nM T25307 C41THR 90203795 IC50 = 14 nM T25307 C4JE9K 90300464 IC50 = 290 nM T25307 CVAW61 90300485 IC50 = 410 nM T25307 C8CBJ5 90305350 IC50 = 6700 nM T25307 CCK2E6 90455013 IC50 = 3.6 nM T25307 CBCE70 90465832 IC50 = 5 nM T25307 CL2R0D 90466288 IC50 = 180 nM T25307 CEB82Q 90646513 Ki = 50 nM T25307 C0Z4BC 90646903 IC50 = 54 nM T25307 C1J5FP 90654865 IC50 = 7560 nM T25307 CP92ZB 90654866 IC50 = 1210 nM T25307 C65MZV 90654867 IC50 = 100 nM T25307 C8JT4Q 90654868 IC50 = 340 nM T25307 C1I7QN 90654869 IC50 = 290 nM T25307 CF1GS0 90654870 IC50 = 2510 nM T25307 C1A6EO 90654871 IC50 = 90 nM T25307 CCAL04 90654872 IC50 = 590 nM T25307 CITM59 90654873 IC50 = 4900 nM T25307 C0O2FD 90654874 IC50 = 410 nM T25307 CR8H6X 90654875 IC50 = 130 nM T25307 CD37WI 90654876 IC50 = 23770 nM T25307 CF4B2A 90654877 IC50 = 52260 nM T25307 CI63QJ 90654878 IC50 = 156300 nM T25307 CA5L3X 90654879 IC50 = 13220 nM T25307 CD6M8S 90654880 IC50 = 174400 nM T25307 CMAD04 90654881 IC50 = 15170 nM T25307 C0K8GI 90654882 IC50 = 2440 nM T25307 C9A8IJ 90654883 IC50 = 9050 nM T25307 CVC05E 90656079 EC50 = 1200 nM T25307 C4DH0F 90656080 EC50 > 10000 nM T25307 CDIE32 90656081 EC50 > 10000 nM T25307 CI8V6K 90656082 EC50 = 360 nM T25307 CD80IL 90656083 EC50 = 1100 nM T25307 CEZ7S9 90656084 EC50 = 3800 nM T25307 C8S9LJ 90656085 IC50 > 10000 nM T25307 C13TEC 90656086 IC50 = 7000 nM T25307 C9FQ2N 90656122 IC50 = 9300 nM T25307 CF4M9V 90656123 IC50 = 6000 nM T25307 C5E6UV 90656124 IC50 = 4200 nM T25307 CS43BG 90656125 IC50 = 1000 nM T25307 C9TI2B 90656126 IC50 = 2600 nM T25307 C35ICO 90656127 IC50 = 4100 nM T25307 CI92WR 91664317 EC50 = 2 nM T25307 CL0GF1 91669190 IC50 = 120 nM T25307 COX5U9 91826672 IC50 = 158.49 nM T25307 CMYL61 91933909 IC50 = 31.62 nM T25307 CXC0M3 92045114 IC50 = 60 nM T25307 C9JFB7 92676534 IC50 = 7510 nM T25307 CFN30K 101783418 EC50 = 1000 nM T25307 CGM78S 117868449 IC50 = 50 nM T25307 CH5F4O 117868534 IC50 = 180 nM T25307 CY72GI 117868652 IC50 = 11 nM T25307 CDZ9S8 117868722 IC50 = 110 nM T25307 CD3C5L 117868794 IC50 = 2000 nM T25307 CF29XT 117868837 IC50 = 2100 nM T25307 CD18IV 117869142 IC50 = 100 nM T25307 CA5DF7 117869398 IC50 = 820 nM T25307 C39JEH 117869438 IC50 = 240 nM T25307 C7ML5B 117869607 IC50 = 21 nM T25307 CC8GN3 117869707 IC50 = 82 nM T25307 CXY6Z8 117869728 IC50 = 5.5 nM T25307 CF69XY 117869774 IC50 = 130 nM T25307 CXTW17 117870010 IC50 = 31 nM T25307 CT3K8B 117940657 EC50 = 47 nM T25307 C9R5HF 117949985 EC50 = 39 nM T25307 C0W6MZ 117950226 EC50 = 32 nM T25307 CYQ36G 117953851 EC50 = 540 nM T25307 CY46RK 117964946 EC50 = 400 nM T25307 CS0G6T 117964950 EC50 = 77 nM T25307 C1WM4V 117964951 EC50 = 220 nM T25307 C2KJH5 117964960 EC50 = 100 nM T25307 C4S9EM 117964962 EC50 = 9 nM T25307 C9AW4X 117964963 EC50 = 670 nM T25307 CS4GJ9 117964973 EC50 = 26 nM T25307 CDXK37 117964975 EC50 = 2 nM T25307 CN6RT8 117964978 EC50 = 10 nM T25307 C0KL3C 117964989 EC50 = 58 nM T25307 C96BSK 117964998 EC50 = 32 nM T25307 C9DK0Q 118005516 IC50 > 6000 nM T25307 COX56L 118005536 EC50 = 49 nM T25307 C9B1SV 118005546 IC50 > 4000 nM T25307 C1UP2D 118005577 IC50 = 310 nM T25307 CNF7K9 118005933 IC50 = 270 nM T25307 C62SPZ 118006087 IC50 = 420 nM T25307 CWJ3B5 118006112 IC50 = 2740 nM T25307 C1O6DM 118006127 IC50 = 200 nM T25307 C7ZV9G 118006189 IC50 > 6000 nM T25307 CP80RJ 118006263 IC50 = 630 nM T25307 C2LCK3 118006433 IC50 = 210 nM T25307 CA1ZP9 118006492 IC50 = 5.3 nM T25307 C0RT5W 118014397 IC50 = 220 nM T25307 C1UN2S 118014429 IC50 = 1900 nM T25307 CA8HX7 118021661 IC50 = 45 nM T25307 CKG0X3 118021909 IC50 = 166 nM T25307 C7BZ3G 118022003 IC50 = 8 nM T25307 C4I0PY 118022053 IC50 = 313 nM T25307 CXF82T 118022242 IC50 = 280 nM T25307 CUJ04F 118022257 IC50 = 2000 nM T25307 CRG8C0 118022267 IC50 = 122 nM T25307 CY27IB 118022286 IC50 = 844 nM T25307 CH4M8W 118022319 IC50 = 193 nM T25307 CEK4F8 118022368 IC50 = 22 nM T25307 CV18BU 118022419 IC50 = 25 nM T25307 C3YT9B 118022425 IC50 = 12 nM T25307 CH6A9O 118022432 IC50 = 29 nM T25307 C1R7KC 118022549 EC50 = 38 nM T25307 C1KAP7 118022609 IC50 = 41 nM T25307 CDJ0S2 118022672 IC50 = 116 nM T25307 CHCI15 118022680 EC50 = 326 nM T25307 C7M0ZH 118022811 IC50 > 6000 nM T25307 CNU54Y 118022821 IC50 = 30 nM T25307 CIL56P 118022829 IC50 = 33 nM T25307 CJF0T8 118022837 IC50 = 20 nM T25307 CD05QE 118022839 IC50 = 19 nM T25307 CO04UZ 118022852 IC50 = 50 nM T25307 CAJU81 118022867 IC50 = 327 nM T25307 CW64FA 118023050 IC50 = 14 nM T25307 C6UG2R 118023068 IC50 = 386 nM T25307 C96LAY 118023081 IC50 = 5.1 nM T25307 CLZV72 118023309 IC50 = 12 nM T25307 CN1M7H 118141954 IC50 = 445 nM T25307 CNM1W9 118141977 IC50 = 37 nM T25307 C56INY 118142016 IC50 = 1.1 nM T25307 CN1LC9 118142017 IC50 = 4 nM T25307 CZ0E5W 118142030 IC50 = 32 nM T25307 C0M8FQ 118142031 IC50 = 205 nM T25307 CW5N0O 118142047 IC50 = 28 nM T25307 C1WA6T 118142048 IC50 = 240 nM T25307 C6IX2E 118142057 IC50 = 140 nM T25307 C96BDN 118142071 IC50 = 29 nM T25307 C1SN3R 118185666 EC50 = 10 nM T25307 CW40HA 118185669 IC50 = 1.6 nM T25307 C2C5KR 118185670 IC50 = 0.69 nM T25307 C8SY3U 118185671 IC50 = 10 nM T25307 CWL6E3 118185675 IC50 = 2.6 nM T25307 C29QXU 118185679 EC50 = 14 nM T25307 CZWL13 118185703 EC50 = 120 nM T25307 CN63GZ 118185705 IC50 = 7.9 nM T25307 CX43PJ 118185706 IC50 = 48 nM T25307 C7KT0M 118185718 IC50 = 0.37 nM T25307 C9AIT5 118185721 IC50 = 1.6 nM T25307 CKT50F 118185722 EC50 = 2.2 nM T25307 CG7FY8 118185723 IC50 = 3.2 nM T25307 CKCO28 118185739 IC50 = 4.4 nM T25307 C01URQ 118185740 IC50 = 21 nM T25307 CI3L8V 118185743 EC50 = 60 nM T25307 C3Z8WU 118185750 IC50 = 33 nM T25307 CMT28E 118185766 IC50 = 0.71 nM T25307 CDB8K3 118185768 IC50 = 20 nM T25307 C1YXL3 118185769 EC50 = 1.3 nM T25307 C0MUP8 118185775 EC50 = 1.6 nM T25307 COH16A 118185777 IC50 = 3.6 nM T25307 C4NM6H 118185785 IC50 = 10 nM T25307 CML8Q4 118186054 EC50 = 60 nM T25307 C4VK9M 118186179 IC50 = 10 nM T25307 C76IFN 118188622 IC50 = 1.4 nM T25307 CDF8G3 118188696 IC50 = 14 nM T25307 C8WXI3 118188704 IC50 = 16 nM T25307 C6WCD0 118188711 EC50 = 12 nM T25307 CIP60N 118188765 IC50 = 7.1 nM T25307 C79IOD 118207841 EC50 = 123 nM T25307 CW27ZE 118207854 IC50 = 146 nM T25307 C2FLM1 118207907 EC50 = 392 nM T25307 CXW5M0 118207954 EC50 = 216 nM T25307 C9UK5A 118207966 EC50 = 128 nM T25307 C0SQH5 118207970 EC50 = 55 nM T25307 C0PWH6 118207991 EC50 = 749 nM T25307 C2U3TJ 118208018 IC50 = 55 nM T25307 C1MOT7 118208026 EC50 = 106 nM T25307 CZ2C3U 118208048 EC50 = 594 nM T25307 CI86YW 118208079 EC50 = 595 nM T25307 C2KAR6 118208086 EC50 = 64 nM T25307 C3TJY2 118208092 EC50 = 4500 nM T25307 CS2F1K 118208112 EC50 = 224 nM T25307 C8N2PF 118208184 EC50 = 36 nM T25307 C9GU8A 118212056 EC50 = 1400 nM T25307 CWO9G0 118212096 EC50 = 232 nM T25307 CKW6P1 118212175 EC50 = 3650 nM T25307 CEU56B 118212311 EC50 = 494 nM T25307 CKU79R 118212564 EC50 = 888 nM T25307 C4DRH0 118212615 EC50 = 271 nM T25307 C51XTL 118217548 EC50 = 378 nM T25307 C1FL5I 118217550 EC50 = 2650 nM T25307 CEN76C 118217555 EC50 = 88 nM T25307 CYRF01 118217561 EC50 = 1040 nM T25307 C2LIW9 118217576 EC50 = 1260 nM T25307 CH9T1O 118217580 EC50 = 4200 nM T25307 CIT31Q 118217593 EC50 = 686 nM T25307 C1ZRN9 118217594 EC50 = 197 nM T25307 CAUT58 118217595 EC50 = 183 nM T25307 CB3KO0 118217596 EC50 = 269 nM T25307 C95ERM 118217608 EC50 = 48 nM T25307 CM2U4C 118217609 EC50 = 61 nM T25307 C9V0ZM 118217611 EC50 = 54 nM T25307 CZ5L3N 118217612 EC50 = 149 nM T25307 CCK3J9 118217851 EC50 = 79 nM T25307 CO5I3V 118217852 EC50 = 508 nM T25307 CD5TJ3 118217853 EC50 = 74 nM T25307 C6HSC3 118217854 EC50 = 31 nM T25307 CEKH57 118217858 EC50 = 33 nM T25307 C1CTB6 118217859 EC50 = 68 nM T25307 C7U0XR 118217863 EC50 = 266 nM T25307 CDP0H5 118217865 EC50 = 590 nM T25307 C82YDU 118217866 EC50 = 1480 nM T25307 CQ60HK 118217867 EC50 = 1260 nM T25307 C9N7VY 118217868 EC50 = 202 nM T25307 C6LC7H 118217869 EC50 = 293 nM T25307 CV9G4S 118217870 EC50 = 572 nM T25307 C8PR3G 118217871 EC50 = 109 nM T25307 CZ3FX6 118217874 EC50 = 1167 nM T25307 CK85HV 118217875 EC50 = 84 nM T25307 CT0DV4 118217911 EC50 = 33 nM T25307 C1QPW5 118217915 EC50 = 129 nM T25307 C3YTM2 118217920 EC50 = 102 nM T25307 CU0T7K 118217922 EC50 = 83 nM T25307 C0ETA2 118217925 EC50 = 146 nM T25307 C89EDG 118217927 EC50 = 161 nM T25307 C81QMJ 118217932 EC50 = 383 nM T25307 C6X4IN 118217935 EC50 = 200 nM T25307 CTNS59 118220706 EC50 = 643 nM T25307 CHY3F8 118220811 EC50 = 1130 nM T25307 CVAL24 118222973 IC50 = 4 nM T25307 CJT5N4 118223005 IC50 = 6.9 nM T25307 C04CPR 118223074 IC50 = 26 nM T25307 CF95US 118223084 IC50 = 410 nM T25307 CM3CW8 118223093 IC50 = 5 nM T25307 CPF3V2 118223167 IC50 = 100 nM T25307 CA8CJ2 118348709 EC50 < 500 nM T25307 CEQ4D3 118348757 EC50 < 500 nM T25307 CZT23F 118395829 IC50 = 316.23 nM T25307 C5DMF9 118395881 IC50 = 50.12 nM T25307 CPZ2J7 118395885 IC50 = 100 nM T25307 C4T5JP 118395947 IC50 = 125.89 nM T25307 C0FO9R 118526820 EC50 = 150 nM T25307 CGX71L 118526824 EC50 = 4500 nM T25307 CD01CA 118526849 EC50 = 27 nM T25307 CY7HP4 118526913 IC50 = 340 nM T25307 CW0GY1 118526919 IC50 = 180 nM T25307 CQL52E 118526951 EC50 = 50 nM T25307 CJ89QH 118526984 IC50 = 14 nM T25307 C15LCG 118526998 IC50 = 21 nM T25307 C75OCQ 118527009 EC50 = 340 nM T25307 C5S6JG 118527010 EC50 = 340 nM T25307 C6GPT5 118527019 EC50 = 240 nM T25307 CM08SP 118622736 IC50 = 2 nM T25307 CX47JR 118658423 IC50 = 110 nM T25307 CN6O2P 118658525 IC50 = 7.5 nM T25307 CQ5Y4W 118658608 IC50 = 200 nM T25307 CEC7A6 118658636 IC50 = 3.9 nM T25307 C2SR9Q 118658701 IC50 = 2.5 nM T25307 C1VGU2 118704903 EC50 = 820 nM T25307 CRN58P 118707352 IC50 = 12000 nM T25307 CZ7M8V 118707353 EC50 = 1000 nM T25307 CZIH01 118707354 EC50 = 13 nM T25307 CZ3JM8 118707355 EC50 = 53 nM T25307 CS3NP5 118707356 EC50 = 1 nM T25307 CILA24 118707357 IC50 = 100 nM T25307 CZI9G0 118707359 EC50 < 50 nM T25307 CUKY97 118708430 EC50 = 20 nM T25307 CC41MJ 118708431 EC50 = 42 nM T25307 CU7VS6 118708432 EC50 > 10000 nM T25307 C7B8SA 118711154 IC50 = 6.5 nM T25307 CIW74L 118724650 EC50 = 1000 nM T25307 CJI3Z8 118724651 IC50 = 66 nM T25307 C9L7GK 118724652 IC50 = 430 nM T25307 CQA30O 118724653 EC50 = 56 nM T25307 CBZ75K 118724654 EC50 = 15 nM T25307 CN7EO3 118728935 IC50 = 5700 nM T25307 C5ZK0R 118728936 IC50 = 4100 nM T25307 C63WOV 118728937 IC50 = 2200 nM T25307 CT85YK 118728938 IC50 = 1900 nM T25307 CVX23H 118728939 IC50 = 1100 nM T25307 C0Q9BW 118728940 IC50 = 440 nM T25307 C69LGI 118728941 IC50 = 1000 nM T25307 CYP4H7 118728942 IC50 = 5600 nM T25307 CWG65E 118728943 IC50 = 16000 nM T25307 CW9VU6 118728944 IC50 = 18000 nM T25307 CJS1C8 118865568 IC50 = 12.8 nM T25307 CBCP16 118865570 IC50 = 7.9 nM T25307 C8KO5R 118865601 IC50 = 638 nM T25307 CB0AH7 118865631 IC50 = 5 nM T25307 C27MYR 118865641 IC50 = 295 nM T25307 CW9U0I 118865660 IC50 = 19.9 nM T25307 CM78FW 118865699 IC50 = 783 nM T25307 C5B8IN 118865703 IC50 = 5 nM T25307 C5HF8A 118977582 IC50 = 14 nM T25307 C92YEL 118977746 IC50 = 4.1 nM T25307 C2Q3VM 118977846 IC50 = 20 nM T25307 C1K2XL 118977850 IC50 = 10 nM T25307 CRU6F4 118987241 IC50 = 56 nM T25307 COT95F 121316232 IC50 = 4.4 nM T25307 C3TWP6 121316298 IC50 = 1.9 nM T25307 CU91LZ 121316306 IC50 = 4.8 nM T25307 C93DUY 121316369 IC50 = 6.4 nM T25307 CU9GE7 121316520 IC50 = 2.5 nM T25307 CV61GY 121316689 IC50 = 300 nM T25307 CK9CN8 121316758 IC50 = 870 nM T25307 CCD3R6 121316759 IC50 = 57 nM T25307 C6TBD2 121345502 EC50 = 34 nM T25307 CS06LH 121345503 EC50 = 2700 nM T25307 C79ARM 121345638 EC50 = 2500 nM T25307 CH4UW8 121345685 EC50 = 11000 nM T25307 C7LRC9 121345693 EC50 = 16000 nM T25307 C9XM0S 121345804 EC50 = 1700 nM T25307 C67JEK 121345817 EC50 = 960 nM T25307 CO45ZP 121345821 EC50 = 13000 nM T25307 CX27VB 121345824 EC50 > 20000 nM T25307 CZQ9R8 121345843 EC50 = 1700 nM T25307 CHWU32 121345862 EC50 = 980 nM T25307 C93FOK 121345869 EC50 > 20000 nM T25307 CI52WN 121345902 EC50 = 2800 nM T25307 CJ1YQ0 121345913 EC50 = 6400 nM T25307 CC13GH 121345920 EC50 = 920 nM T25307 C0AUP8 121345965 EC50 > 20000 nM T25307 C2UZ1V 121346049 EC50 = 3900 nM T25307 C70XUF 121346140 EC50 = 230 nM T25307 CQ7M9L 121346161 EC50 = 2900 nM T25307 C34RDH 121346173 EC50 = 900 nM T25307 C3GK7I 121346194 EC50 > 20000 nM T25307 C7ZW4R 121346196 EC50 = 1300 nM T25307 CC63UM 121346198 EC50 = 6700 nM T25307 CUIP05 121346222 EC50 = 440 nM T25307 CR5VK1 121346230 EC50 = 1800 nM T25307 C0A1XC 121414058 IC50 = 210 nM T25307 C1MTH5 121414062 IC50 = 34 nM T25307 CM0L6H 121414081 IC50 = 6400 nM T25307 CPZ0W3 121414092 IC50 = 610 nM T25307 C9TE3S 121414113 IC50 = 390 nM T25307 C2KOJ9 121414123 IC50 = 97 nM T25307 CGDQ80 121414138 IC50 = 490 nM T25307 CKG61D 121414144 IC50 = 44 nM T25307 C5TEX7 121414150 IC50 = 68 nM T25307 CV1N3J 121414174 IC50 = 1100 nM T25307 COSM18 121414176 IC50 = 690 nM T25307 CY1ZJ4 121414177 IC50 = 30 nM T25307 CPSZ82 121429360 IC50 = 89 nM T25307 C82UPO 121429364 IC50 = 220 nM T25307 C1KZ5U 121429459 IC50 > 10000 nM T25307 C4OB7L 121429472 IC50 = 320 nM T25307 C04LCM 121429512 IC50 = 86 nM T25307 C7D3AT 121429517 IC50 = 17 nM T25307 CFTS73 121429519 IC50 = 47 nM T25307 C2JGN3 121429520 IC50 = 20 nM T25307 CV5R4G 121470704 IC50 = 1 nM T25307 C85HZL 121470706 IC50 = 2 nM T25307 C09QGL 121470709 IC50 = 37 nM T25307 C3OL2H 121480641 IC50 = 11 nM T25307 CD89ZC 121480642 IC50 = 25 nM T25307 CO6HF9 122180196 IC50 = 5500 nM T25307 CIX4M5 122180197 IC50 = 5400 nM T25307 C2YWB1 122180198 IC50 = 4200 nM T25307 CEW72J 122180199 IC50 = 4400 nM T25307 CLR57W 122182699 EC50 = 97 nM T25307 CPJ3M7 122182700 EC50 = 840 nM T25307 CK5WJ9 122182701 EC50 = 190 nM T25307 CY0M6P 122182702 EC50 = 250 nM T25307 CLV91R 122182703 EC50 = 240 nM T25307 CIZG84 122182883 IC50 = 7100 nM T25307 C03NCQ 122182884 EC50 = 484 nM T25307 CRIZ31 122182885 EC50 = 101 nM T25307 C4SGV6 122182886 IC50 = 10 nM T25307 CEK2R7 122182887 IC50 = 3 nM T25307 CP71OW 122182888 IC50 = 710 nM T25307 C5L1AS 122184114 EC50 = 49 nM T25307 CUC7A1 122184123 EC50 = 12 nM T25307 CLZU40 122184130 EC50 = 71 nM T25307 CP0V1K 122184132 EC50 = 150 nM T25307 CL7EY2 122184139 EC50 = 13 nM T25307 CE87BY 122184140 EC50 = 10 nM T25307 CGQW03 122184141 EC50 > 1000 nM T25307 C6M7TB 122184142 EC50 > 1000 nM T25307 CHUW19 122184171 EC50 = 84 nM T25307 CC2GS5 122184172 EC50 = 2600 nM T25307 CM3IU2 122184173 EC50 > 10000 nM T25307 C1UG6Y 122184174 EC50 > 10000 nM T25307 CI4WF2 122184175 EC50 > 10000 nM T25307 CS23CB 122184176 EC50 = 6800 nM T25307 CFMX82 122184177 EC50 = 440 nM T25307 C5VH7R 122186246 IC50 = 1995.26 nM T25307 C1WJH2 122186247 IC50 = 2511.89 nM T25307 CP1AC3 122186248 EC50 = 15.85 nM T25307 CR2TM7 122187573 IC50 = 7943.28 nM T25307 CZ9R8H 122187574 IC50 = 398.11 nM T25307 CSHD85 122187575 IC50 = 79.43 nM T25307 C9XPA8 122187576 IC50 > 25118.86 nM T25307 CW6L5E 122187577 IC50 = 501.19 nM T25307 CKFG83 122187578 IC50 > 25118.86 nM T25307 CI43GD 122187579 IC50 = 501.19 nM T25307 C4JF6M 122187580 IC50 = 158.49 nM T25307 CEMD59 122187581 IC50 = 6.31 nM T25307 CRY8N5 122190169 EC50 = 86 nM T25307 CJ97KI 122190170 EC50 = 230 nM T25307 CA24WF 122190171 EC50 > 10000 nM T25307 C5QCI3 122190172 EC50 > 10000 nM T25307 CB9GP5 122235238 IC50 = 40 nM T25307 C0WAM1 122379290 EC50 = 47 nM T25307 CID82P 122644619 EC50 = 13 nM T25307 C4F9ZK 122669103 EC50 = 19 nM T25307 CZH39M 122669106 EC50 = 7 nM T25307 C0T8FO 122669173 EC50 = 15 nM T25307 CD6X5P 122669265 EC50 = 24 nM T25307 C0S7UB 122678562 EC50 = 35 nM T25307 CY8S1P 122678563 EC50 = 21 nM T25307 C0MUW2 122678576 EC50 = 8 nM T25307 C2SQ9M 122678748 EC50 = 16 nM T25307 CH1J6K 122678779 EC50 = 16 nM T25307 CD9HN3 122678983 EC50 = 17 nM T25307 CF39TE 122679031 EC50 = 150 nM T25307 C41GNL 124374661 IC50 = 3980 nM T25307 CXRL40 126599968 IC50 = 4 nM T25307 CRU2V4 127028566 IC50 = 10 nM T25307 CBDV53 127028567 IC50 = 72 nM T25307 CUK1L6 127028568 IC50 = 72 nM T25307 C95VHK 127029741 IC50 = 200 nM T25307 C0XWI7 127029952 IC50 = 11000 nM T25307 CY9X5C 127029953 IC50 > 30000 nM T25307 C80JHT 127029994 IC50 = 520 nM T25307 C7X0VL 127031148 EC50 = 450 nM T25307 C6B5EQ 127031440 EC50 > 20000 nM T25307 CMF87T 127032960 EC50 = 9500 nM T25307 C5BJY6 127033009 EC50 = 850 nM T25307 C0QP2N 127046061 IC50 = 10430 nM T25307 CQ12BK 127046268 IC50 = 22050 nM T25307 CRYO71 127046810 IC50 = 770 nM T25307 C49VCF 127046811 IC50 = 11290 nM T25307 CI1RP7 127047257 IC50 = 220 nM T25307 CRU15Q 127047258 IC50 = 10320 nM T25307 C85SAR 127047259 IC50 = 25830 nM T25307 CR0Y1J 127047260 IC50 = 630 nM T25307 C1EY6K 127047332 IC50 = 13600 nM T25307 C2Y3KM 127047492 IC50 = 3650 nM T25307 C9YAT2 127047774 IC50 = 67050 nM T25307 C14KQI 127048039 IC50 = 112250 nM T25307 C4W7VR 127048040 IC50 = 620 nM T25307 CWM97P 127048041 IC50 = 1310 nM T25307 CIT35Z 127048042 IC50 = 910 nM T25307 C1UY2C 127053200 IC50 = 4200 nM T25307 CY1D9H 127053204 IC50 = 1500 nM T25307 CCIK23 127053205 IC50 = 3800 nM T25307 CB0MV9 127053206 IC50 = 3200 nM T25307 CLM5V7 127053207 IC50 > 10000 nM T25307 CJ0W2M 127053208 IC50 = 4700 nM T25307 CGQ94Y 127053209 IC50 = 7800 nM T25307 C8XD0P 127053213 IC50 = 210 nM T25307 C3OT0Z 127053216 IC50 = 910 nM T25307 CN0HD3 127053223 IC50 > 10000 nM T25307 C2WJN3 127053224 IC50 = 10000 nM T25307 C47LWE 127053237 IC50 = 520 nM T25307 CT0UB3 127053238 IC50 = 2800 nM T25307 C75GOB 127053239 IC50 = 630 nM T25307 CE3MI7 127053240 IC50 = 6500 nM T25307 C2P8QB 127053243 IC50 > 10000 nM T25307 CQM6F2 127053244 IC50 = 6400 nM T25307 C8JW1U 129167185 EC50 = 280 nM T25307 CD2LP9 130248006 IC50 = 3460 nM T25307 CXUK13 130261792 IC50 = 820 nM T25307 CNA0D8 130261824 IC50 = 1080 nM T25307 C0S5RN 130261825 IC50 = 930 nM T25307 C4BGQ0 130261871 IC50 = 1980 nM T25307 CB8IS1 130261967 IC50 = 7660 nM T25307 CHON78 130262004 IC50 = 1830 nM T25307 C31FOZ 130262014 IC50 = 4170 nM T25307 CM3NE7 130262015 IC50 = 1490 nM T25307 C9NVI7 130262024 IC50 = 3080 nM T25307 C4L1PC 130262081 IC50 = 1490 nM T25307 CO7DT9 130262256 IC50 = 1520 nM T25307 CR91VO 130262355 IC50 = 7550 nM T25307 CL8QD5 130262897 IC50 = 8050 nM T25307 CZCU47 130262898 IC50 = 8720 nM T25307 CXD2F4 130262938 IC50 = 4240 nM T25307 CJG42F 130263340 IC50 = 2220 nM T25307 C17WQM 130263494 IC50 = 460 nM T25307 C5ZXU2 130263507 IC50 = 7760 nM T25307 CDV84X 131747741 EC50 = 9 nM T25307 CKT8C5 131747744 EC50 = 7 nM T25307 CW18DI 131747749 EC50 = 17 nM T25307 CK53XU 131747768 EC50 = 12 nM T25307 CB62QX 131953519 EC50 = 12 nM T25307 C1CR0K 132274777 EC50 = 19.95 nM T25307 CZU10O 132473003 EC50 = 25.12 nM T25307 C7CZG3 134131811 IC50 = 2700 nM T25307 CP1U5T 134132295 IC50 = 120 nM T25307 CB6C7O 134133110 IC50 > 10000 nM T25307 C2Z0DR 134133677 IC50 > 10000 nM T25307 C0VX8Q 134135363 IC50 = 1200 nM T25307 C1UVG3 134137057 IC50 = 260 nM T25307 C60HIA 134137870 IC50 > 10000 nM T25307 CGO9C7 134138123 IC50 = 300 nM T25307 CH9VS2 134138409 IC50 = 2600 nM T25307 CL85MU 134139004 IC50 = 6200 nM T25307 CK5CZ8 134139028 IC50 = 310 nM T25307 CR7J9Q 134139617 IC50 > 10000 nM T25307 CJQ8O6 134139787 IC50 = 3600 nM T25307 CH4O7X 134140416 IC50 = 370 nM T25307 C7TMP3 134140572 IC50 = 54 nM T25307 CR0CX8 134141317 IC50 = 820 nM T25307 C5Y0XG 134141341 IC50 = 6500 nM T25307 CS4V8O 134141363 IC50 > 10000 nM T25307 C61WKA 134142331 IC50 = 88 nM T25307 CR69NQ 134142378 IC50 = 3600 nM T25307 C8FS0G 134142941 IC50 = 4300 nM T25307 CKD1S2 134144175 IC50 > 10000 nM T25307 C8QNS0 134145062 IC50 > 10000 nM T25307 C4AO0F 134145297 IC50 = 2500 nM T25307 CCWS64 134145922 IC50 > 10000 nM T25307 C68HUB 134146033 IC50 = 2500 nM T25307 C6XZY1 134147284 IC50 > 10000 nM T25307 CY4R8J 134147557 IC50 > 10000 nM T25307 C3AHY8 134147641 IC50 > 10000 nM T25307 C9LPU5 134148070 IC50 = 6000 nM T25307 CLC9U8 134148522 IC50 = 1200 nM T25307 CT6GX8 134148836 IC50 > 10000 nM T25307 CV1MC9 134149320 IC50 = 5900 nM T25307 C07QGW 134149538 IC50 = 9200 nM T25307 CJ75KB 134149807 IC50 = 5000 nM T25307 CPO31X 134150617 IC50 = 1100 nM T25307 COC3J0 134151576 IC50 > 10000 nM T25307 CO12JS 134152058 IC50 = 4800 nM T25307 C0MNC7 134152441 IC50 = 720 nM T25307 CC30KS 134153013 IC50 > 10000 nM T25307 C6B5DW 134154628 IC50 = 1800 nM T25307 CHIZ89 134155284 IC50 = 590 nM T25307 C3PGZ2 134155420 IC50 = 2100 nM T25307 C8HJE4 134156268 IC50 = 4800 nM T25307 CTV56P 134156567 IC50 > 10000 nM T25307 CVER01 134157830 IC50 > 10000 nM T25307 CX27TP 134693870 IC50 = 255 nM T25307 C2ZMU3 134812586 IC50 = 20 nM T25307 C7KI8H 134812587 IC50 = 20 nM T25307 CG6H3K 134812588 IC50 = 19 nM T25307 CK0Y6M 134812713 IC50 = 14 nM T25307 C9FKU2 134817202 IC50 = 420 nM T25307 CB3HG0 134817247 IC50 = 9 nM T25307 C4TPN6 134821990 IC50 = 14 nM T25307 CMS25F 135133967 IC50 = 290 nM T25307 CR2BH6 135133982 IC50 = 81 nM T25307 C30NHW 137387862 EC50 = 18 nM T25307 CE8W9L 137399015 IC50 = 3000 nM T25307 C19OIK 137399020 IC50 = 81.9 nM T25307 C46JFK 137399564 IC50 = 1450 nM T25307 CP8SX4 137399571 IC50 = 1100 nM T25307 CIT2C3 137399640 IC50 = 69.6 nM T25307 CCV9A6 137399832 IC50 = 566 nM T25307 C2M9HO 137399842 IC50 = 156 nM T25307 C2PT9G 137399843 IC50 = 58.5 nM T25307 CK9OW5 137399857 IC50 = 1220 nM T25307 CKJW86 137400175 IC50 = 54.9 nM T25307 CFU52C 137400227 IC50 = 167 nM T25307 C9YX4Z 137400228 IC50 = 5400 nM T25307 C4BGZ9 137400229 IC50 = 138 nM T25307 CQ1I0Z 137641042 IC50 = 3 nM T25307 CU0W5I 137642486 IC50 = 3 nM T25307 C69JNL 137646533 IC50 = 3.2 nM T25307 CK3X1N 137796283 IC50 = 13 nM T25307 CSY2G3 138105957 IC50 = 30 nM T25307 CEZY91 138115387 IC50 = 14 nM T25307 C1KV0T 138393322 IC50 = 44 nM T25307 CM6OB9 138454290 IC50 = 50.12 nM T25307 C03DMN 138654637 IC50 = 10 nM T25307 CB98IG 138697431 IC50 = 2960 nM T25307 COS34U 138698013 IC50 = 90 nM T25307 CHW10Q 138805804 IC50 = 17 nM T25307 C72TYC 139035058 EC50 = 20.8 nM T25307 CP02YQ 140430650 IC50 = 29 nM T25307 CFG46S 140430651 IC50 = 5 nM T25307 C3YWI4 140430652 IC50 = 21 nM T25307 C37JUM 140773958 IC50 = 46 nM T25307 C73RKI 140774004 IC50 = 7.6 nM T25307 CX6R0A 140774032 IC50 = 17 nM T25307 CWO2E7 140774044 IC50 = 4.2 nM T25307 CY3VR7 140774049 IC50 = 3.8 nM T25307 CGIB87 140774080 IC50 = 3.5 nM T25307 CU3G1E 140774123 IC50 = 24 nM T25307 C6PFG8 140774153 IC50 = 4.1 nM T25307 CK61GB 140774194 IC50 = 4.5 nM T25307 C6KXU3 140774249 IC50 = 3.1 nM T25307 C3O7JB 140781127 IC50 = 110 nM T25307 COWE15 140781228 IC50 = 57 nM T25307 CXFE08 140781243 IC50 = 48 nM T25307 CBL73J 140781279 IC50 = 160 nM T25307 CUMI75 140941226 IC50 = 7.8 nM T25307 CJ2R7W 141493565 EC50 = 8 nM T25307 C7XT6D 141493567 EC50 = 3 nM T25307 C9WMS8 141738698 IC50 = 313 nM T25307 C1LJ8X 141738716 IC50 = 47.8 nM T25307 CFO03M 141738729 IC50 = 426 nM T25307 CO4J6W 141738741 IC50 = 358 nM T25307 CE20XR 141761791 IC50 = 960 nM T25307 CBV6F5 141761792 IC50 = 2280 nM T25307 CKM8L4 141761793 IC50 = 4160 nM T25307 CC2BH9 145232219 IC50 < 30 nM T25307 CF96VY 145714275 IC50 = 117.5 nM T25307 CW3Y0H 145949340 IC50 > 20000 nM T25307 CL61DH 145950915 IC50 = 75 nM T25307 C6U2NZ 145951285 IC50 = 14 nM T25307 CI7PN5 145951364 IC50 = 3250 nM T25307 CLR1U4 145951408 IC50 = 40 nM T25307 CEG51M 145951461 IC50 = 88 nM T25307 CY0IK8 145951714 IC50 = 59 nM T25307 CIDZ65 145951873 IC50 = 7 nM T25307 CQK8E9 145952014 IC50 = 3.1 nM T25307 CYQ7M2 145952483 IC50 = 1146 nM T25307 C9DMC6 145952803 IC50 = 66 nM T25307 CIX31H 145952816 EC50 = 39.81 nM T25307 C7E4BV 145952831 IC50 = 440 nM T25307 C02ADZ 145953181 IC50 = 46 nM T25307 CEKV06 145953371 IC50 = 30 nM T25307 CUY6A2 145953373 IC50 = 79.43 nM T25307 CC89ZA 145954089 IC50 = 4900 nM T25307 CDQK14 145954301 IC50 = 2 nM T25307 CZ47LO 145954717 IC50 = 50 nM T25307 CRY37A 145954889 IC50 = 780 nM T25307 C48FJG 145955283 IC50 = 9000 nM T25307 CYS80W 145955432 IC50 = 700 nM T25307 CIGS39 145955613 IC50 = 23 nM T25307 C67MPG 145955616 IC50 = 144 nM T25307 C0P5BV 145955708 IC50 = 18 nM T25307 C1YXC2 145955835 IC50 = 80 nM T25307 CQH7E1 145956869 IC50 = 20 nM T25307 C4WIZ9 145956958 IC50 = 770 nM T25307 CR70ZO 145957041 IC50 = 49 nM T25307 CUZC01 145957673 EC50 = 125.89 nM T25307 C8IS2U 145957844 IC50 > 10000 nM T25307 C60CMX 145958026 IC50 = 7 nM T25307 C3PQ5Y 145958747 IC50 = 31.62 nM T25307 CGIE51 145958813 IC50 = 27 nM T25307 COX51S 145959004 IC50 = 50.12 nM T25307 CL2HT7 145959111 IC50 = 3 nM T25307 C07PAH 145959487 IC50 = 110 nM T25307 CXFC59 145959683 IC50 = 30 nM T25307 CEYP23 145959816 IC50 = 100 nM T25307 CX70MO 145959855 IC50 = 125.89 nM T25307 CR38GE 145960090 IC50 = 15000 nM T25307 CYC64Q 145960155 IC50 = 25 nM T25307 C91KPX 145960248 IC50 = 19 nM T25307 C3AQ6L 145961003 IC50 = 120 nM T25307 CE61YH 145961343 IC50 = 6.1 nM T25307 CIMW18 145961622 IC50 = 1.8 nM T25307 CMGC52 145961772 IC50 = 2.6 nM T25307 CR2SG1 145961853 IC50 = 29 nM T25307 CJ7RU8 145961892 IC50 = 1 nM T25307 CP2N3K 145962172 IC50 = 1.3 nM T25307 C56QRW 145962236 IC50 = 209 nM T25307 CWRU80 145962336 IC50 = 9.4 nM T25307 C6ZLK4 145962447 IC50 = 43 nM T25307 CEU4V3 145962457 IC50 = 4.7 nM T25307 CN7Z3Q 145963286 EC50 = 317 nM T25307 C01QZJ 145963443 IC50 = 6.3 nM T25307 CR7GX1 145963554 IC50 = 17 nM T25307 CZM2D7 145963820 EC50 = 195 nM T25307 C9AT7Y 145964005 EC50 > 10000 nM T25307 CKJI71 145964066 IC50 = 7670 nM T25307 C2AP9V 145964523 EC50 = 165 nM T25307 CN25FE 145964574 IC50 > 50000 nM T25307 CI3TP7 145964673 EC50 = 225 nM T25307 CIE7J6 145965097 IC50 = 6600 nM T25307 CFK0H4 145965098 EC50 = 203 nM T25307 CKL63D 145965344 EC50 = 1640 nM T25307 C13SNC 145965495 EC50 = 15 nM T25307 C3GI6D 145965669 EC50 = 114 nM T25307 C4TL7G 145965870 EC50 = 84 nM T25307 C9GF1S 145965986 IC50 = 99 nM T25307 CQ5UT9 145965987 EC50 = 230 nM T25307 C4H9UY 145966156 EC50 = 165 nM T25307 CJ1T7B 145966372 IC50 > 30000 nM T25307 CEVT16 145966599 IC50 = 7200 nM T25307 CQ7W5N 145966640 EC50 = 530 nM T25307 CJ0H3D 145966902 EC50 = 2040 nM T25307 C4P3DR 145967002 EC50 = 240 nM T25307 C4O7RB 145967121 IC50 = 7.5 nM T25307 CQFI17 145967205 IC50 = 5700 nM T25307 CK4W1H 145967316 IC50 = 5160 nM T25307 CO02AH 145967656 IC50 > 40000 nM T25307 CTUC50 145967755 IC50 = 5.3 nM T25307 C4JZ8T 145967902 IC50 > 40000 nM T25307 C3PZ8R 145967947 IC50 = 39 nM T25307 CY9M6W 145968047 IC50 = 6300 nM T25307 CY1X5Q 145968478 EC50 = 2780 nM T25307 CKT3A4 145968585 IC50 > 40000 nM T25307 C2EU7Y 145968591 IC50 = 5500 nM T25307 CYS1Z3 145968983 IC50 = 6800 nM T25307 CBQ91G 145968987 IC50 > 40000 nM T25307 CHDX94 145969211 IC50 = 4400 nM T25307 C0GX6M 145969292 IC50 = 13400 nM T25307 C76RKW 145969356 IC50 > 40000 nM T25307 CG27VL 145969403 EC50 = 80 nM T25307 CX7GL1 145970040 IC50 > 40000 nM T25307 C05RUB 145970465 IC50 = 260 nM T25307 CFK76Y 145970594 IC50 > 40000 nM T25307 C2IU3H 145970596 IC50 = 840 nM T25307 C67OZA 145970683 IC50 = 2300 nM T25307 CGR9U4 145970687 IC50 = 16100 nM T25307 CV1EB9 145971091 IC50 = 6500 nM T25307 CPJI78 145971170 IC50 > 40000 nM T25307 CYT8M9 145971562 EC50 = 31 nM T25307 CB96HZ 145971912 IC50 > 10000 nM T25307 C1L8QS 145972171 IC50 = 17 nM T25307 CR0Z5S 145972196 IC50 = 6000 nM T25307 C3L8WH 145973447 IC50 = 16200 nM T25307 CC8HN9 145973516 EC50 = 28 nM T25307 CZO15G 145973599 IC50 = 69000 nM T25307 C0X3EB 145974156 EC50 = 15 nM T25307 CE91FN 145974227 IC50 = 230 nM T25307 C21ERW 145974493 IC50 = 75 nM T25307 C13TQJ 145974494 EC50 = 170 nM T25307 CFH2G9 145974751 IC50 = 2.8 nM T25307 CAYQ72 145974767 EC50 = 93 nM T25307 C8J3WE 145974803 IC50 = 60 nM T25307 C3QHV8 145974820 IC50 = 6 nM T25307 C0QKU3 145975648 EC50 = 170 nM T25307 C60CDE 145975835 EC50 = 7500 nM T25307 CA3XR1 145976113 EC50 = 58 nM T25307 C1G0IJ 145976189 IC50 = 1320 nM T25307 CS5IH8 145976365 IC50 = 84 nM T25307 CM98RL 145976534 EC50 > 10000 nM T25307 CQZ7I9 145977465 EC50 = 600 nM T25307 CO50LX 145977718 EC50 < 500 nM T25307 CE2O1P 145977892 EC50 = 815 nM T25307 C9UTC7 145977974 IC50 = 914 nM T25307 CEXF68 145978063 IC50 = 35 nM T25307 CQ7GS8 145978084 EC50 > 10000 nM T25307 CA4X9J 145978153 IC50 > 30000 nM T25307 C6SQ9I 145978824 EC50 = 1260 nM T25307 CD37PO 145979241 IC50 = 10700 nM T25307 C49DSL 145979648 IC50 = 3800 nM T25307 CVZ07E 145979726 IC50 = 9.8 nM T25307 CEX6U7 145979878 IC50 = 40 nM T25307 C8AF9R 145980027 IC50 < 30 nM T25307 CB70AE 145980094 IC50 = 16 nM T25307 CD57NU 145980245 IC50 = 7.6 nM T25307 C6XD5G 145980263 IC50 = 25 nM T25307 CR7XF1 145980684 IC50 = 4.8 nM T25307 CBC03Q 145981346 IC50 < 30 nM T25307 CW7M6O 145981666 IC50 = 40 nM T25307 CXE1L6 145981784 IC50 < 30 nM T25307 CS7UC0 145981807 IC50 = 1800 nM T25307 C3XFE9 145981969 IC50 = 11 nM T25307 CXW29A 145982397 IC50 = 2900 nM T25307 C5VBU6 145982695 IC50 = 1000 nM T25307 C1JUC8 145982712 IC50 = 56 nM T25307 C8G4QR 145982788 IC50 > 30000 nM T25307 C3OI9S 145983415 IC50 = 277 nM T25307 CU0V8B 145984255 IC50 > 30000 nM T25307 C9XWV7 145984603 IC50 > 30000 nM T25307 CYRX35 145985210 IC50 > 30000 nM T25307 CP9Q8O 145985306 IC50 > 30000 nM T25307 C89ZMA 145985638 IC50 > 40000 nM T25307 CX27GB 145985841 IC50 = 63 nM T25307 C7UD5H 145985845 IC50 = 30 nM T25307 C4S0VC 145986574 IC50 = 170 nM T25307 C8R1PL 145986833 IC50 = 64 nM T25307 CK9E7I 145987745 IC50 = 4700 nM T25307 CRTG03 145987785 IC50 = 25 nM T25307 C4JSI1 145987881 IC50 = 33 nM T25307 CF0K5O 145987907 IC50 < 30 nM T25307 CAU45I 145987980 IC50 > 3000 nM T25307 C8C5KF 145988118 IC50 = 3800 nM T25307 CI6H1L 145988123 IC50 = 31 nM T25307 CM0G9W 145988515 IC50 > 5000 nM T25307 CM2WR3 145988768 IC50 = 36 nM T25307 C4ESM8 145988957 IC50 = 460 nM T25307 CDI01N 145989245 IC50 = 790 nM T25307 C4RQW3 145989261 IC50 = 71 nM T25307 CWSP97 145989563 IC50 = 2600 nM T25307 CX5BG3 145989591 IC50 = 15 nM T25307 C7HGR2 145989697 IC50 = 6800 nM T25307 CN7V5K 145989867 IC50 = 242 nM T25307 CE47TS 145990013 IC50 = 4.4 nM T25307 CH0W7O 145990222 IC50 = 310 nM T25307 C1FOL5 145990361 IC50 = 97 nM T25307 CG02OC 145990362 IC50 > 5000 nM T25307 C8DUV3 145990929 IC50 = 150 nM T25307 C4W7IA 145991126 IC50 = 330 nM T25307 CC4DV9 145991246 IC50 = 780 nM T25307 C0Q8PC 145991576 IC50 = 36 nM T25307 CY58DQ 145991674 IC50 = 10000 nM T25307 CFK69N 145992026 IC50 = 8.2 nM T25307 CUM7Z6 145992194 IC50 = 64 nM T25307 C0EB5D 145992591 IC50 = 14000 nM T25307 CDR1L5 145992630 IC50 = 28 nM T25307 C8R2QA 145992708 IC50 = 49 nM T25307 C3Q0ZN 145993067 IC50 = 14000 nM T25307 C4VYJ2 145993264 IC50 = 67 nM T25307 CNKZ14 145993272 IC50 = 140 nM T25307 C29-APR 145993797 IC50 = 20 nM T25307 C09XNT 145994167 IC50 = 500 nM T25307 CGXM06 146673074 IC50 = 51 nM T25307 CC89OI 148034311 EC50 = 9 nM T25307 C4ZR9N 148795928 EC50 = 19000 nM T25307 CHAN48 150802389 IC50 = 44 nM T25307 CNRW91 154641330 EC50 = 43.6 nM T25307 CXN0T4 154649064 IC50 = 1090 nM T25307 CMG2U5 154649065 IC50 = 6620 nM T25307 C6JG4B 154649067 IC50 = 30900 nM T25307 CR6C2G 154649070 IC50 = 1750 nM T25307 C7DJ9Z 154649071 IC50 > 100000 nM T25307 CHYI48 154649073 IC50 = 9600 nM T25307 CB0WU5 155007664 IC50 = 62600 nM T25307 CPTL34 155491026 IC50 > 100000 nM T25307 CUFS62 155510496 EC50 = 6 nM T25307 CE90TC 155510591 EC50 = 9.5 nM T25307 C71TPI 155510740 EC50 = 25.5 nM T25307 C9K7HE 155511006 IC50 = 25.12 nM T25307 CVP75I 155511045 IC50 = 128 nM T25307 C89IPO 155511076 EC50 = 31.1 nM T25307 CE6V8Z 155511797 EC50 = 43 nM T25307 CKQ1B2 155511896 IC50 = 264.9 nM T25307 C56XWT 155512000 IC50 = 91100 nM T25307 CKY9S4 155513376 EC50 = 205 nM T25307 C0XF2E 155513913 IC50 = 569.3 nM T25307 CN4H2V 155513917 IC50 = 464.9 nM T25307 CI2W0G 155514259 EC50 = 42.6 nM T25307 C7VO4K 155514401 EC50 = 244 nM T25307 C34VBF 155514962 IC50 = 251 nM T25307 CPNW63 155515051 EC50 = 87.4 nM T25307 C9J0HG 155515245 EC50 = 50.6 nM T25307 C8KBQ6 155515430 IC50 = 1692.5 nM T25307 C8T2YZ 155515472 IC50 = 384.7 nM T25307 C27FUT 155515808 IC50 = 3200 nM T25307 CY7F5P 155516459 IC50 = 39.81 nM T25307 CL21PV 155516814 IC50 = 70 nM T25307 C98SLC 155516898 IC50 = 1674.5 nM T25307 C15CTM 155516899 IC50 = 6149 nM T25307 C7ID2S 155517084 IC50 = 53500 nM T25307 CH56FO 155517423 IC50 = 111 nM T25307 CS93NA 155517530 IC50 = 12.59 nM T25307 CE8R2A 155517869 IC50 = 79.43 nM T25307 CM3B0N 155518095 IC50 = 4 nM T25307 C3D2VX 155518209 EC50 = 2.1 nM T25307 C30SPO 155518654 IC50 = 25 nM T25307 C18KMV 155518729 IC50 = 14 nM T25307 CQJX03 155519864 IC50 = 36 nM T25307 C8TH4B 155520423 EC50 = 4.1 nM T25307 C5P3EX 155520776 IC50 = 199 nM T25307 CJKZ61 155521375 EC50 = 39.3 nM T25307 CJ70LO 155521467 IC50 = 63.1 nM T25307 CO2DV5 155521917 EC50 = 74.3 nM T25307 C9WJN5 155522706 IC50 = 399.9 nM T25307 CU5Z8T 155522788 EC50 = 42 nM T25307 CVK29S 155522978 EC50 = 133 nM T25307 C7IDH0 155523063 IC50 = 210 nM T25307 C9JL6O 155523070 IC50 = 8760 nM T25307 C2DO9Y 155523351 IC50 = 73900 nM T25307 CSQ82C 155523503 EC50 = 47.9 nM T25307 C5OV8D 155523841 IC50 = 5 nM T25307 CK0R1I 155523977 IC50 = 290 nM T25307 CJZ36P 155524235 IC50 = 251.19 nM T25307 CC2L9J 155524508 EC50 = 56.8 nM T25307 C3T4EL 155524825 IC50 = 6 nM T25307 C5B8HJ 155524925 EC50 = 45.3 nM T25307 C5O0PA 155525359 IC50 = 158.49 nM T25307 CUP65T 155525416 IC50 = 5575 nM T25307 CDS84A 155525533 IC50 > 100000 nM T25307 C1DT9M 155525669 EC50 = 270 nM T25307 CO93DB 155525763 IC50 = 925.1 nM T25307 C6S5JG 155526041 EC50 = 21.8 nM T25307 C1F8OC 155526216 IC50 = 130 nM T25307 C1I5QF 155526863 EC50 = 124 nM T25307 C7Y5ZR 155526875 IC50 = 3.162 nM T25307 C8N9XS 155526930 EC50 = 16.1 nM T25307 CXS9T8 155526989 EC50 = 10 nM T25307 CGU6T4 155527039 EC50 = 14.6 nM T25307 C1TIY2 155528097 EC50 = 93.8 nM T25307 CBZ6O7 155528556 EC50 = 52.3 nM T25307 C5X9KL 155528844 EC50 = 209 nM T25307 C19XSN 155528909 IC50 = 124 nM T25307 CSY9V5 155529269 IC50 = 107 nM T25307 CEP5X0 155529423 IC50 > 1000 nM T25307 CUAY47 155529665 IC50 = 125.89 nM T25307 C2HEC1 155530220 IC50 = 50.12 nM T25307 CW30ZF 155530247 IC50 = 1589.5 nM T25307 CDC8R1 155530281 IC50 = 93 nM T25307 CWDX63 155530392 IC50 = 8410 nM T25307 CW89HU 155530658 EC50 = 11 nM T25307 CO9N5H 155530678 EC50 = 29 nM T25307 CQIJ85 155530797 EC50 = 99.4 nM T25307 C4IHK3 155531439 EC50 = 286 nM T25307 C9BMT1 155531456 IC50 = 5 nM T25307 CM0QV8 155532208 IC50 = 158 nM T25307 C21KSE 155532294 IC50 > 100000 nM T25307 CY0M8V 155532844 IC50 = 50.12 nM T25307 C0LS3V 155533208 EC50 = 41.3 nM T25307 CA87YX 155533211 IC50 = 39.81 nM T25307 C5M2GZ 155533435 IC50 = 153.7 nM T25307 C94HPY 155533857 EC50 = 31.3 nM T25307 CI24FJ 155534295 IC50 = 213 nM T25307 CZD65G 155534599 IC50 = 63.1 nM T25307 CCEH31 155534678 IC50 = 79 nM T25307 CCY96X 155534713 IC50 = 2442.5 nM T25307 CZ0C7B 155534979 EC50 = 78.8 nM T25307 CG7R3B 155535010 IC50 = 1900 nM T25307 CHQ7C4 155535342 IC50 = 20 nM T25307 CTI4O7 155535733 IC50 = 8000 nM T25307 CBK01J 155536039 IC50 = 230 nM T25307 CPL38V 155536831 IC50 = 207.9 nM T25307 CI3O4K 155537342 IC50 = 873.4 nM T25307 CF9I3X 155537626 IC50 = 39.81 nM T25307 CIUA10 155537856 EC50 = 13 nM T25307 CCO96S 155538113 IC50 = 20 nM T25307 C4TU1Y 155538306 IC50 = 18 nM T25307 CZ41RY 155538359 IC50 = 366.7 nM T25307 CW7EK5 155538714 IC50 = 1574.5 nM T25307 C07BZT 155538928 IC50 = 333.2 nM T25307 CLO98T 155539150 EC50 = 56 nM T25307 COP7X8 155539171 IC50 = 70 nM T25307 CK4W7I 155539903 IC50 = 1512.5 nM T25307 CE9XL7 155541551 EC50 = 2 nM T25307 C7Q1FJ 155541575 IC50 > 100000 nM T25307 C8YA3R 155541656 EC50 = 106 nM T25307 CMIT24 155542434 IC50 = 15.85 nM T25307 C92OWA 155542651 EC50 = 6 nM T25307 C10FEH 155542743 IC50 = 10000 nM T25307 CPDU07 155542796 EC50 = 125 nM T25307 C0V6EY 155543172 EC50 = 12 nM T25307 CS8Y4O 155543462 IC50 = 350 nM T25307 CRWD76 155544210 EC50 = 26.2 nM T25307 CR8E1D 155544300 IC50 = 717.9 nM T25307 C1DYL0 155544357 EC50 = 1300 nM T25307 CX7L0S 155544387 EC50 = 16 nM T25307 CSK20E 155544524 EC50 = 7 nM T25307 CTEC81 155544796 EC50 = 396 nM T25307 CVE05C 155545976 EC50 = 230 nM T25307 CSFQ34 155546436 EC50 = 57.1 nM T25307 CZ05OD 155546712 IC50 = 1200 nM T25307 CCQ7D5 155547247 IC50 = 48 nM T25307 CRSO75 155547762 IC50 = 830 nM T25307 C1U8PB 155548703 EC50 = 80.4 nM T25307 CK2WY8 155548972 IC50 = 2010 nM T25307 CZMQ20 155549008 IC50 = 290 nM T25307 CHN46C 155549055 IC50 = 9 nM T25307 C7TG3I 155549124 EC50 = 120 nM T25307 CO5VN7 155549587 EC50 = 30.2 nM T25307 CEJP15 155549607 EC50 = 43.4 nM T25307 CM0KR4 155550145 IC50 = 4897.5 nM T25307 CPV48H 155550250 IC50 = 240 nM T25307 CYQ24A 155550306 IC50 = 50.12 nM T25307 C4N7TL 155550468 IC50 = 8242 nM T25307 C5V6ZQ 155551512 EC50 = 25.2 nM T25307 C0MBP5 155551516 EC50 = 6 nM T25307 CS9CW8 155552387 IC50 > 10000 nM T25307 CM73VP 155552403 IC50 = 506 nM T25307 CHS09K 155553079 IC50 = 1500 nM T25307 CVFB83 155553194 IC50 = 288.4 nM T25307 CM2SU0 155553245 EC50 = 820 nM T25307 C5C4PI 155553279 EC50 = 94 nM T25307 C8IXR7 155553715 EC50 = 122 nM T25307 CC98VB 155553746 IC50 = 287.2 nM T25307 C7N5HA 155554052 IC50 = 38 nM T25307 C05WBK 155554057 EC50 = 8 nM T25307 CR3WG9 155554123 EC50 = 25.7 nM T25307 CUEH60 155554280 IC50 = 105 nM T25307 C50AZQ 155554971 EC50 = 31 nM T25307 CDK3O4 155555014 IC50 = 21 nM T25307 CF1D4A 155555172 IC50 = 39.81 nM T25307 CQTJ01 155555204 EC50 = 8 nM T25307 CX19JM 155555274 IC50 > 10000 nM T25307 CB1Z2J 155555405 IC50 = 8.1 nM T25307 C64QRM 155555952 IC50 = 59 nM T25307 CBK1E5 155556708 EC50 = 17 nM T25307 CQB48L 155556931 IC50 = 15 nM T25307 C5LTZ2 155557446 IC50 = 93 nM T25307 CN08CY 155557709 IC50 = 590 nM T25307 C8P9LU 155558273 EC50 = 28 nM T25307 CIZT32 155558566 IC50 = 10 nM T25307 C7OTA5 155559009 EC50 = 1900 nM T25307 C61QGX 155559146 EC50 = 410 nM T25307 CBR4Z7 155559595 EC50 = 32.9 nM T25307 C6HN5D 155559896 IC50 = 270.3 nM T25307 C9CSL1 155559954 IC50 = 50 nM T25307 CUP04O 155560017 IC50 = 4 nM T25307 CKWX81 155560289 EC50 = 3800 nM T25307 C3FI7U 155560819 EC50 = 20 nM T25307 CF72VK 155560886 EC50 = 7 nM T25307 C2MIY4 155560987 IC50 > 3000 nM T25307 C74ASN 155561045 EC50 = 410 nM T25307 C4S9AD 155561084 IC50 > 100000 nM T25307 CF8LU0 155561764 EC50 = 58 nM T25307 CUN8D9 155561950 IC50 = 3 nM T25307 CO4VK0 155561972 IC50 = 21 nM T25307 C1ZIR7 155562040 EC50 = 42 nM T25307 CNSG86 155562159 IC50 > 10000 nM T25307 CN1LS2 155563358 IC50 = 41 nM T25307 CMT5Z9 155563591 EC50 = 73 nM T25307 C7DMU4 155563611 EC50 = 21 nM T25307 C64KEH 155564120 EC50 = 3900 nM T25307 CHP6S0 155564297 EC50 = 7 nM T25307 CIBA72 155564665 IC50 = 16 nM T25307 CA91EM 155564933 EC50 = 23 nM T25307 CPF42S 155565257 EC50 = 10 nM T25307 CW41YG 155565880 IC50 = 4 nM T25307 CRSL75 155566131 IC50 = 79.43 nM T25307 C59EOG 155566503 EC50 = 34 nM T25307 CX7GO4 155567273 IC50 = 23 nM T25307 CH26TK 155567292 IC50 = 193.6 nM T25307 CYD8T9 155567508 EC50 = 7 nM T25307 CJ32AZ 155567529 IC50 = 75 nM T25307 CXM4R3 155567816 EC50 = 49.3 nM T25307 C43LBV 155567951 IC50 = 156 nM T25307 CC1X2G 155569065 IC50 = 357.7 nM T25307 C5GXM4 155569310 IC50 = 27 nM T25307 CI1ML2 155569453 EC50 > 10000 nM T25307 C7W1YC 118707360 EC50 < 100 nM T25307 CO6A4S 122184103 IC50 = 240 nM T25307 CA36YE 122184104 EC50 = 1700 nM T25307 CK05OP 122184105 IC50 = 38 nM T25307 CA3F5R 122184106 EC50 = 1200 nM T25307 CIA3T6 122184107 EC50 = 160 nM T25307 C6KMU5 122184108 IC50 = 18 nM T25307 C2MEG0 122184109 IC50 = 76 nM T25307 CYOP26 122184110 EC50 = 130 nM T25307 CV5CO0 122184112 IC50 = 8.6 nM T25307 C63QAO 122184113 IC50 = 3.8 nM T25307 CT3WD4 122184116 EC50 = 6.1 nM T25307 CBHT23 122184117 IC50 = 4.8 nM T25307 CH1EJ7 122184118 EC50 = 33 nM T25307 CGD7W0 122184119 EC50 = 22 nM T25307 CW7Z3Q 122184120 EC50 = 14 nM T25307 CGTV80 122184121 EC50 = 7.6 nM T25307 CSAQ70 122184122 EC50 = 15 nM T25307 C9CWU6 122184124 EC50 = 15 nM T25307 CW05RP 122184125 IC50 = 70 nM T25307 CQ57GP 122184126 EC50 = 25 nM T25307 C2FGW1 122184127 IC50 = 16 nM T25307 CX3UB0 122184128 EC50 = 21 nM T25307 CQ3E4C 122184129 EC50 = 37 nM T25307 CXP8Q3 122184131 IC50 = 21 nM T25307 C13QFC 122184133 EC50 = 9.5 nM T25307 CAR25O 122184134 EC50 = 13 nM T25307 CS3DB5 122184135 EC50 = 55 nM T25307 C4H3NW 122184136 EC50 = 76 nM T25307 CO82BL 122184137 EC50 = 12 nM T25307 CPM90L 122184138 EC50 = 17 nM T25307 D01RNA 439577 EC50 = 80 nM T25307 D02DLW 5997 EC50 = 20 nM T25307 D02RQP 6623 IC50 > 10000 nM T25307 D06OVX 65094 EC50 = 20 nM T25307 D07LUJ 64945 IC50 = 130 nM T25307 D08URT 121948 Ki = 10 nM T25307 D0B5FC 447912 Ki = 51 nM T25307 D0FB7S 473141 Ki = 10 nM T25307 D0G6JM 5289501 EC50 = 9000 nM T25307 D0K4GK 167685 EC50 = 20 nM T25307 D0K5QH 107722 Ki = 10 nM T25307 D0O1WJ 44241473 Ki = 111 nM T08280 D0R9OH 5329 IC50 > 57000 nM T08280 D0H2UB 5361 IC50 = 3000 nM T08280 C67KIW 1010711 IC50 = 14600 nM T08280 CZS7X1 1290388 IC50 = 1830 nM T08280 CGB7V9 2431573 IC50 = 410 nM T08280 C96AMV 2434603 IC50 > 57000 nM T08280 CIMO36 2678352 IC50 = 79 nM T08280 C2RIJ9 5220784 IC50 = 36600 nM T08280 C47SDJ 22829926 IC50 = 16300 nM T08280 C85FYO 25014723 IC50 = 23000 nM T08280 CID0O3 44585245 IC50 = 50000 nM T08280 CQDP20 44585248 IC50 = 80000 nM T08280 C0ON3R 44585364 IC50 = 49000 nM T08280 C8Q9BZ 44585399 IC50 = 410000 nM T08280 CQ90ZU 46871719 IC50 = 30000 nM T08280 C0HY2U 46891355 IC50 = 170000 nM T08280 CUS8Z2 46891410 Ki = 10000 nM T08280 C0CJU2 53255376 IC50 = 6510 nM T08280 C2SMU5 53255377 IC50 = 5800 nM T08280 CT7P0Y 53255378 IC50 = 7300 nM T08280 CL9SV8 53255380 IC50 = 33000 nM T08280 C3HDS6 53255382 IC50 = 1460 nM T08280 CMIF14 53255383 IC50 = 680 nM T08280 CFME61 53255385 IC50 = 5170 nM T08280 C9AV6I 53255391 IC50 > 57000 nM T08280 C27BLC 53255392 IC50 = 112 nM T08280 CE9R2J 53255393 IC50 = 520 nM T08280 CJA02O 53255401 IC50 = 2310 nM T08280 C83ZQN 53255402 IC50 = 16300 nM T08280 CA8U6N 53255404 IC50 = 2590 nM T08280 CCY4S2 53255406 IC50 > 57000 nM T08280 CJU24X 53255407 IC50 = 820 nM T08280 C8BM2S 53255416 IC50 > 57000 nM T08280 CFQS86 53255418 IC50 = 260 nM T08280 C8HMA5 53255419 IC50 = 4610 nM T08280 C2LN4A 53255421 IC50 = 370 nM T08280 C1F5NM 53255422 IC50 > 57000 nM T08280 CCK76U 53255423 IC50 = 36600 nM T08280 CF73JM 53255425 IC50 = 160 nM T08280 CRD14K 53255426 IC50 = 6000 nM T08280 CL6X3U 53255427 IC50 = 6510 nM T08280 C0RI7V 53255428 IC50 = 730 nM T08280 C7E2CW 53255430 IC50 = 700 nM T08280 C6EY3P 53255432 IC50 = 5800 nM T08280 CK59IB 53255434 IC50 = 18300 nM T08280 C9IM0N 53255435 IC50 = 37000 nM T08280 CQ0E3W 53255437 IC50 = 650 nM T08280 CC0U9P 53255438 IC50 = 2910 nM T08280 CWM1K7 53255440 IC50 = 5160 nM T08280 C1X2HV 53255442 IC50 = 32600 nM T08280 C2FKX6 73670805 IC50 = 15 nM T08280 CNP40G 76335640 IC50 = 24 nM T08280 C8WRY1 90666782 IC50 = 900000 nM T08280 CQ5EF3 90666783 IC50 = 410000 nM T08280 D0M5KC 46871703 Ki = 9000 nM T98078 CP6VN4 2328332 IC50 = 6626 nM T98078 CW54IK 3781024 IC50 = 3361 nM T98078 C1JLR8 4610393 IC50 = 930 nM T98078 CU1MB3 9868957 IC50 = 22 nM T98078 C3BQ8I 9924885 IC50 = 41 nM T98078 C80RKE 9969262 IC50 = 460 nM T98078 CSH4E2 10110611 IC50 = 19.95 nM T98078 CS6BG9 10111090 IC50 = 95 nM T98078 CRM59T 10114592 IC50 = 79 nM T98078 CLTE80 10116214 IC50 = 730 nM T98078 CLW0T7 10117032 IC50 = 9 nM T98078 CS3T9V 10131968 IC50 = 407.38 nM T98078 C38PHC 10132088 IC50 = 0.85 nM T98078 C5RFN0 10133605 IC50 = 0.29 nM T98078 CDJ56V 10134098 IC50 = 288.4 nM T98078 CIU29K 10137647 IC50 = 2770 nM T98078 C5MTH3 10138012 IC50 = 1200 nM T98078 CU93YP 10138176 IC50 = 1300 nM T98078 CTX32H 10140171 IC50 = 2550 nM T98078 C6Y4WR 10140239 IC50 = 251.19 nM T98078 CW91ZC 10140861 IC50 = 53.7 nM T98078 C0TS9M 10144673 IC50 = 11 nM T98078 CSY9E5 10155073 IC50 = 680 nM T98078 C5BS7H 10156838 IC50 = 650 nM T98078 C0QN3M 10158463 IC50 = 990 nM T98078 CG92QM 10160614 IC50 = 26 nM T98078 C5HFB4 10161428 IC50 = 31 nM T98078 C4VLG2 10164669 IC50 = 416.87 nM T98078 CZ3X4P 10177786 IC50 = 1130 nM T98078 CVA6K1 10178588 IC50 = 137 nM T98078 CRMX64 10178913 IC50 = 960 nM T98078 C70LPF 10178967 IC50 = 1160 nM T98078 C92ZBW 10179150 IC50 = 34 nM T98078 C6NL8B 10181847 IC50 = 19 nM T98078 CU3XB9 10184715 IC50 = 2970 nM T98078 C5FN2V 10199888 IC50 = 670 nM T98078 C5G0JH 10200929 IC50 = 70.79 nM T98078 CX8L3I 10206413 IC50 = 41.69 nM T98078 C1OGD3 10207019 IC50 = 389.05 nM T98078 CZ94LH 10221600 IC50 = 630 nM T98078 C7W3KU 10223147 IC50 = 31 nM T98078 C5IM3Y 10225184 IC50 = 40 nM T98078 CBN34A 10226392 IC50 = 1480 nM T98078 CD2UA5 10227245 IC50 = 338.84 nM T98078 CD7V6Z 10269568 IC50 = 0.98 nM T98078 CBC73I 10270539 IC50 = 28 nM T98078 C0X3ER 10270978 IC50 = 60 nM T98078 C4RSN8 10271223 IC50 = 1990 nM T98078 CT96UE 10271742 IC50 = 1 nM T98078 CIE89F 10271802 IC50 = 1780 nM T98078 C3N0ZS 10272000 IC50 = 930 nM T98078 CNU17W 10272495 IC50 = 190 nM T98078 CTID39 10273201 IC50 = 34 nM T98078 CV3Z0M 10273363 IC50 = 37 nM T98078 C6NL5H 10274098 IC50 = 20 nM T98078 CAK4L6 10274153 IC50 = 30.2 nM T98078 C0AS5Z 10277212 IC50 = 42.66 nM T98078 COCS61 10294500 IC50 = 2540 nM T98078 C1OX8N 10296234 IC50 = 8 nM T98078 C59TWR 10297307 IC50 = 389.05 nM T98078 CA1K9U 10297689 IC50 = 19.95 nM T98078 CY8S1Z 10299006 IC50 = 14 nM T98078 C8Y4AE 10387489 IC50 = 23 nM T98078 C36DNE 11501492 IC50 = 1767 nM T98078 C5WRZ6 11503947 IC50 = 580 nM T98078 CD85AQ 11510695 IC50 = 5 nM T98078 C63NWA 11524152 IC50 = 1147 nM T98078 CSGZ61 11525705 IC50 = 75 nM T98078 CR65TN 11525725 IC50 = 150 nM T98078 CIS2U1 11530524 IC50 = 1.14 nM T98078 C3V2PO 11531889 IC50 = 10 nM T98078 C7T1ZS 11532776 IC50 = 45 nM T98078 CN3CE4 11539051 IC50 = 5 nM T98078 CYHE92 11539363 IC50 = 7 nM T98078 CP1J7Z 11545653 IC50 = 28 nM T98078 CKF0Z5 11546160 IC50 = 165.96 nM T98078 CFK20O 11546847 IC50 = 376 nM T98078 C1RT6O 11553802 IC50 = 199 nM T98078 CWDZ52 11577040 IC50 = 37 nM T98078 CE9S6K 11581962 IC50 = 421 nM T98078 CA97VB 11582572 IC50 = 168 nM T98078 CGO8Z4 11582784 IC50 = 60 nM T98078 C48BXR 11583513 IC50 = 30 nM T98078 C6ADC9 11595890 IC50 = 106 nM T98078 C2I1JM 11597257 IC50 = 17 nM T98078 CSBM48 11602463 IC50 = 801 nM T98078 CISJ92 11604132 IC50 = 175 nM T98078 CY3AE9 11610826 IC50 = 2.65 nM T98078 CY32EU 11612176 IC50 = 7.943 nM T98078 CI3W8L 11612369 IC50 = 105 nM T98078 CC2N6J 11618087 IC50 = 28 nM T98078 CNJ2G8 11625482 IC50 = 74 nM T98078 C43ALZ 11626431 IC50 = 245.47 nM T98078 CMS1R4 11632456 IC50 = 627 nM T98078 CK6JA9 11632811 IC50 = 1.99 nM T98078 C0I3DS 11632812 IC50 = 773 nM T98078 C2DO8U 11634442 IC50 = 269 nM T98078 CS9O4R 11639462 IC50 = 1015 nM T98078 CVO0E9 11640826 IC50 = 80 nM T98078 C0SK3F 11641706 IC50 = 9 nM T98078 CHM49J 11646151 IC50 = 59 nM T98078 CZR2X4 11646266 IC50 = 489 nM T98078 CFT52G 11646592 IC50 = 463 nM T98078 C6KH3X 11647479 IC50 = 8 nM T98078 CAG38C 11647480 IC50 = 136 nM T98078 CAHG23 11653196 IC50 = 676 nM T98078 CI18ZL 11655768 IC50 = 72.44 nM T98078 CNW83Q 11661015 IC50 = 321 nM T98078 CTC91X 11674345 IC50 = 1.45 nM T98078 C4XTP1 11674573 IC50 = 177.83 nM T98078 CYZ5D6 11677029 IC50 = 15 nM T98078 C4REG1 11683974 IC50 = 99 nM T98078 C23LRG 11689700 IC50 = 1564 nM T98078 CFH83T 11710602 IC50 = 394 nM T98078 CN92XI 11711262 IC50 = 20 nM T98078 CZH02U 11711494 IC50 = 7 nM T98078 C4B2YC 11712118 IC50 = 140 nM T98078 CJ3T6W 11712783 IC50 = 113 nM T98078 CZ80HK 11718085 IC50 = 4337 nM T98078 CM7HT9 16721146 IC50 = 68 nM T98078 CHX6A5 25023822 IC50 = 2298 nM T98078 CM9ON6 44333328 IC50 = 13.3 nM T98078 CPW58N 44407162 IC50 = 74000 nM T98078 CMQC96 44407163 IC50 = 58.88 nM T98078 CFK6D9 44407166 IC50 = 340000 nM T98078 CXWE57 44407171 IC50 = 302 nM T98078 CB1W5T 44407172 IC50 = 482000 nM T98078 C01TEM 44407197 IC50 = 3730 nM T98078 COVD95 44407198 IC50 = 116 nM T98078 C7FE8Y 44407199 IC50 = 190.55 nM T98078 C3F5UZ 44407200 IC50 = 316.23 nM T98078 C0VB8E 44407204 IC50 = 341000 nM T98078 CA06UW 44407205 IC50 = 140 nM T98078 C8XDV0 44407206 IC50 = 567000 nM T98078 C59NJP 44407207 IC50 = 243000 nM T98078 CRP5D8 44407211 IC50 = 20000 nM T98078 C21ZOW 44407212 IC50 = 55000 nM T98078 CQP0W2 44407225 IC50 = 3160 nM T98078 CJKG07 44407231 IC50 = 147.91 nM T98078 C4A5LS 44407236 IC50 = 200 nM T98078 CB20KF 44407239 IC50 = 4980 nM T98078 CZRJ61 44407240 IC50 = 791000 nM T98078 CJM2P8 44407241 IC50 = 107000 nM T98078 CS06NA 44407243 IC50 = 168 nM T98078 C9XFB2 44407257 IC50 = 523000 nM T98078 CRIC04 44407260 IC50 = 467.74 nM T98078 CM5J1B 44407261 IC50 = 321000 nM T98078 C3O7HW 44407262 IC50 = 274000 nM T98078 C4BRK2 44407263 IC50 = 114 nM T98078 CSU4H5 44407264 IC50 = 1080000 nM T98078 CR18CA 44407267 IC50 = 65 nM T98078 C7LZE2 44407278 IC50 = 37 nM T98078 CL3BS9 44407279 IC50 = 239.88 nM T98078 CFD76L 44407280 IC50 = 223.87 nM T98078 CYJK38 44407286 IC50 = 163000 nM T98078 C3P2RH 44407287 IC50 = 5320 nM T98078 CNF80D 44407288 IC50 = 87.1 nM T98078 CFB98S 44407289 IC50 = 41 nM T98078 C1SVA0 44407290 IC50 = 3330 nM T98078 CK43YM 44413236 IC50 = 3332 nM T98078 C07BTJ 44413237 IC50 = 112.2 nM T98078 CC8V9W 44413318 IC50 = 148 nM T98078 CHY45C 44413319 IC50 = 47 nM T98078 CS6L9Z 44413320 IC50 = 117 nM T98078 C5VCY9 44413331 IC50 = 438 nM T98078 CM25HV 44413332 IC50 = 1280 nM T98078 C2PX6G 44413337 IC50 = 235 nM T98078 CQTW62 44413338 IC50 = 84 nM T98078 CVHC51 44413350 IC50 = 353 nM T98078 C52IMF 44413351 IC50 = 1576 nM T98078 C2URO0 44413419 IC50 = 24 nM T98078 C9QF8L 44413431 IC50 = 794 nM T98078 CN2F5Q 44413432 IC50 = 984 nM T98078 CU2D7J 44413433 IC50 = 22 nM T98078 CZ7K9M 44413448 IC50 = 1711 nM T98078 CE78FH 44413449 IC50 = 689 nM T98078 CI5E6J 44413450 IC50 = 187 nM T98078 CVJ46K 44413451 IC50 = 356 nM T98078 C5BRD2 44413485 IC50 = 177.83 nM T98078 CH27FY 44413486 IC50 = 526 nM T98078 C05AVE 44438394 IC50 = 5450 nM T98078 C2YZ0B 44438395 IC50 = 4900 nM T98078 CE1K9M 44438396 IC50 = 1500 nM T98078 CX59TV 44438397 IC50 = 4500 nM T98078 CLM75P 44438398 IC50 = 17200 nM T98078 C95BLI 44438399 IC50 = 2800 nM T98078 CTNO30 44438401 IC50 = 1731 nM T98078 C49EUM 44438403 IC50 = 151.36 nM T98078 CK43QJ 44438405 IC50 = 80 nM T98078 C2QA9I 44438406 IC50 = 73 nM T98078 CJ3TH2 44438407 IC50 = 1531 nM T98078 CDV42I 44438408 IC50 = 2034 nM T98078 CSXL18 44438409 IC50 = 679 nM T98078 C4I6XP 44438410 IC50 = 115 nM T98078 C6VD2F 44438414 IC50 = 239.88 nM T98078 C0CN8S 44438415 IC50 = 2753 nM T98078 C9JP2H 44438416 IC50 = 302 nM T98078 CUA65D 44438422 IC50 = 5011 nM T98078 CQ8M9N 44438425 IC50 = 507 nM T98078 CYX0S7 44438426 IC50 = 654 nM T98078 CAB3P0 44438427 IC50 = 1739 nM T98078 C5CTL6 44438428 IC50 = 1351 nM T98078 CF46IT 44438429 IC50 = 562.34 nM T98078 CFE1L5 44438430 IC50 = 953 nM T98078 CJ8L2U 44438431 IC50 = 154.88 nM T98078 CL0TP2 44438433 IC50 = 214 nM T98078 CZN3F8 44438434 IC50 = 399 nM T98078 C4QFJ2 44438435 IC50 = 1105 nM T98078 C0ZXC4 44438437 IC50 = 1619 nM T98078 C0LEX9 44438438 IC50 = 3280 nM T98078 CG4P0A 44445017 IC50 = 154.88 nM T98078 CJ47KV 44445019 IC50 = 118 nM T98078 C4AM7W 44445020 IC50 = 208.93 nM T98078 CSOW09 44445021 IC50 = 44 nM T98078 C89BMW 44445026 IC50 = 346.74 nM T98078 C3H6IS 46208235 IC50 = 2.3 nM T98078 C8TA9V 49800128 IC50 = 4.9 nM T98078 CB7OP1 52940749 IC50 = 110 nM T98078 C95GPY 52940787 IC50 = 46 nM T98078 C9C2YE 52940984 IC50 = 1.4 nM T98078 C69ZDF 52941309 IC50 = 19 nM T98078 CZ3WR6 52941362 IC50 = 0.6 nM T98078 C1X7GW 52941384 IC50 = 1.7 nM T98078 CF01QR 52941425 IC50 = 240 nM T98078 CR59NK 52941432 IC50 = 12 nM T98078 CG4T5K 52941433 IC50 = 3.3 nM T98078 COKB09 52941546 IC50 = 2.2 nM T98078 C7JF0P 52941934 IC50 = 3.1 nM T98078 C49LZX 52942525 IC50 = 14 nM T98078 CYQ54H 52942570 IC50 = 11 nM T98078 CAO42E 52942713 IC50 = 6.7 nM T98078 CAU1N9 52942806 IC50 = 1.6 nM T98078 CLO2U4 52943200 IC50 = 1.1 nM T98078 C6LXS4 52943360 IC50 = 8.7 nM T98078 CG51JU 52943361 IC50 = 4.7 nM T98078 C4V3GP 52943769 IC50 = 13 nM T98078 CW7QK8 52943794 IC50 = 20 nM T98078 CR49TW 52943918 IC50 = 2.7 nM T98078 C0Q7VT 52944048 IC50 = 19 nM T98078 CR4A1P 52944059 IC50 = 24 nM T98078 C5VT6P 52944118 IC50 = 8.9 nM T98078 C1QIN4 52944347 IC50 = 4.5 nM T98078 CV6KG2 52944549 IC50 = 79 nM T98078 C97UDC 52944582 IC50 = 1.6 nM T98078 CE2A5B 52944895 IC50 = 37 nM T98078 CGY24R 52944985 IC50 = 0.5 nM T98078 CY2Z9I 52945062 IC50 = 4 nM T98078 C5LW7Q 52945148 IC50 = 5.7 nM T98078 CVKN95 52946280 IC50 = 1.8 nM T98078 C5LW9X 52946339 IC50 = 16 nM T98078 C42MBW 52948260 IC50 = 8.1 nM T98078 CRVZ90 52948685 IC50 = 0.9 nM T98078 CP0L4A 52948966 IC50 = 11 nM T98078 CW2LN6 52948988 IC50 = 92 nM T98078 CS2TV3 52948994 IC50 = 5.1 nM T98078 C6ZD3Y 52949260 IC50 = 59 nM T98078 CU4S5E 52949298 IC50 = 76 nM T98078 CT1JF3 52949520 IC50 = 11 nM T98078 CCD0Z7 52949786 IC50 = 36 nM T98078 C4OD8Q 52949870 IC50 = 44 nM T98078 CEC6R8 52949929 IC50 = 320 nM T98078 CW3Z5I 52949933 IC50 = 0.9 nM T98078 CY1A8J 52949976 IC50 = 42 nM T98078 CYT6Z8 52949994 IC50 = 3.2 nM T98078 CA8F9B 52949995 IC50 = 600 nM T98078 COB13J 52949996 IC50 = 450 nM T98078 CV9F4D 52950006 IC50 = 1.3 nM T98078 C6KOB4 135453421 IC50 = 1170 nM T47594 D06TFI 10090485 IC50 = 199 nM T47594 D0E3TC 44259 IC50 = 9118 nM T47594 D0MR0B 54766013 IC50 = 13 nM T47594 D0T3ME 156422 IC50 = 44000 nM T47594 CD4Y0N 11682470 IC50 = 46 nM T47594 C7YG1N 24759534 IC50 = 200 nM T47594 CPQ31L 25195294 IC50 = 1825 nM T47594 CN2QG1 44223357 IC50 = 1840 nM T47594 C3VRO9 44557921 IC50 > 10000 nM T47594 CDV74N 50997747 IC50 = 9622 nM T47594 C0SWH5 53348216 IC50 > 40000 nM T47594 C8NA4L 53384644 IC50 = 35000 nM T47594 C6EIN3 56663574 IC50 = 882 nM T47594 COKW25 56666809 IC50 = 224 nM T47594 C7CID9 56667031 IC50 = 108 nM T47594 C0OE8R 56677286 IC50 = 18 nM T47594 C4X0FD 56683923 IC50 = 956 nM T47594 CXJ63M 59603829 IC50 = 170 nM T47594 CQEU96 59603842 IC50 = 730 nM T47594 CIP7B1 60182373 IC50 = 3420 nM T47594 CQ6KV9 60182388 IC50 = 4090 nM T47594 CK6WO0 66552478 IC50 < 10000 nM T47594 C91RWL 66561650 IC50 = 59 nM T47594 C5DGR9 69036886 IC50 = 10000 nM T47594 C1HW4B 89735655 IC50 > 100000 nM T47594 C2LD1B 121232401 IC50 = 31 nM T47594 C9CV7H 121411850 IC50 < 100 nM T47594 CU3BI0 121412063 IC50 < 100 nM T47594 CI2YE9 132606873 IC50 = 2761 nM T47594 CPT0V7 138454752 IC50 = 18330 nM T47594 C2MD1Q 155513187 IC50 > 10000 nM T47594 D05NEC 60182364 IC50 = 183 nM T47594 D0C3AD 10202642 IC50 > 1000 nM T47594 D0F2MP 60182389 IC50 = 326 nM T47594 D0K6YK 11676119 IC50 = 23 nM T47594 D0PP6Y 60182393 IC50 = 5930 nM T47594 D0Q5UH 9858940 IC50 = 70 nM T47594 D0Y0BK 11524144 IC50 = 25740 nM T53748 D00CSQ 5564 Ki = 0.0019 nM T53748 D04AIT 5280445 IC50 = 2000 nM T53748 D0K8KX 5280343 Ki = 22 nM T53748 D0U2BH 65064 Ki = 8 nM T53748 CRB9I1 8468 IC50 = 920000 nM T53748 CTK25Q 72277 Ki = 17.56 nM T53748 CNIW58 107905 Ki = 16 nM T53748 CX52GK 161830 IC50 > 100 ug.mL-1 T53748 CDZ65K 199472 IC50 = 500 nM T53748 CD3U7A 324097 IC50 > 100 ug.mL-1 T53748 CF0C7Y 1202264 IC50 > 100000 nM T53748 CN41BW 1230203 IC50 = 870 nM T53748 C6XQH3 1232811 IC50 > 100000 nM T53748 CJ9K5P 1252780 IC50 = 870 nM T53748 C1YNG2 1268564 Ki = 510 nM T53748 C95LTW 1339021 IC50 = 28500 nM T53748 CZL57W 1355042 Ki = 2000 nM T53748 CP5N1C 1369932 Ki = 880 nM T53748 COH82J 1378575 Ki = 8700 nM T53748 CQP1F8 1382809 IC50 > 100000 nM T53748 CY3V0R 1382811 IC50 > 100000 nM T53748 C3NTJ0 1394341 Ki = 4100 nM T53748 C48ALI 1397803 Ki = 480 nM T53748 CFY3S9 1417792 IC50 = 870 nM T53748 C9Q4MJ 1526752 IC50 = 50000 nM T53748 CO5H2Z 1556190 IC50 > 100000 nM T53748 CL7F2Y 1559978 IC50 > 100000 nM T53748 CFTK12 1560554 IC50 > 100000 nM T53748 CG2O1Z 1561390 IC50 > 100000 nM T53748 C92WGP 1561418 IC50 > 100000 nM T53748 C7ZQ3S 1590532 IC50 > 50000 nM T53748 C81NCI 1718573 IC50 > 100000 nM T53748 CRYH35 1726124 IC50 > 100000 nM T53748 CBV04C 1731052 IC50 = 35000 nM T53748 C81CQX 1839047 IC50 = 25000 nM T53748 CPF89M 1922463 IC50 = 870 nM T53748 CT57VS 2203761 IC50 = 30250 nM T53748 C1EWI3 2244241 Ki = 4.2 nM T53748 C0ER5X 2248987 IC50 > 100000 nM T53748 C0ZAC3 3637765 IC50 = 90000 nM T53748 CX4T5V 4053176 IC50 = 50000 nM T53748 C9T2CI 4391438 IC50 = 52000 nM T53748 C03RFS 4984348 IC50 = 60000 nM T53748 C4SIA8 5280637 IC50 = 10 ug.mL-1 T53748 CY27DM 5283639 IC50 = 18 ug.mL-1 T53748 CKIQ01 5710615 IC50 = 45000 nM T53748 C4NF7P 5710617 IC50 > 100000 nM T53748 C5WTZ8 5710620 Ki = 5100 nM T53748 CNT7K1 5710622 Ki = 6600 nM T53748 C20RNY 5757816 IC50 > 50000 nM T53748 COZ6G0 5759815 IC50 = 20000 nM T53748 CUA07C 5760122 IC50 > 100000 nM T53748 CW54QZ 5847109 IC50 = 1500 nM T53748 C5OS4F 6000620 IC50 > 100000 nM T53748 C0E5OJ 6504827 IC50 = 870 nM T53748 CS95WV 6523040 IC50 > 100000 nM T53748 CP05JD 6524174 IC50 = 870 nM T53748 CL60XC 6914565 IC50 = 310 nM T53748 CJN71Y 6914566 IC50 = 250 nM T53748 CT02JR 6973832 IC50 > 100000 nM T53748 CJTN57 10820593 IC50 > 100 ug.mL-1 T53748 C54AOF 11084315 IC50 = 100 ug.mL-1 T53748 CP59LR 11495355 IC50 = 9000 nM T53748 C8G7VR 11659169 IC50 = 120 nM T53748 CDKE72 11660481 IC50 = 140 nM T53748 C1EL5R 11674015 IC50 = 57 nM T53748 CW06ML 11948630 IC50 = 27000 nM T53748 CP4EW9 16220129 IC50 = 700 nM T53748 C7EG3N 16220130 IC50 = 640 nM T53748 CS76TF 16427167 IC50 > 100000 nM T53748 CY1CK6 17252735 IC50 = 75000 nM T53748 CV51XL 17252838 IC50 = 55000 nM T53748 CAKE96 22427741 IC50 = 60000 nM T53748 CCPJ43 23656593 IC50 > 100000 nM T53748 C1CNR2 25023956 IC50 > 100000 nM T53748 C50SPV 25023957 IC50 = 21000 nM T53748 C5MRD9 25023964 IC50 = 530 nM T53748 CBT9R1 25023965 IC50 = 410 nM T53748 C08NDM 25023970 IC50 = 33000 nM T53748 CT8K9O 25023971 IC50 = 2800 nM T53748 CAG1S3 25023972 IC50 = 840 nM T53748 C4YC3M 25023973 IC50 = 530 nM T53748 CJ35XN 44405271 IC50 = 3000 nM T53748 C96VAD 44405274 IC50 = 460 nM T53748 C8NA5M 44405275 IC50 = 810 nM T53748 C3YR5V 44405276 IC50 = 680 nM T53748 CG6KQ3 44405287 IC50 = 370 nM T53748 C5SY0U 44405289 IC50 = 590 nM T53748 C02SFQ 44405291 IC50 = 200 nM T53748 CR6CE9 44405293 IC50 = 170 nM T53748 C40BRH 44405298 IC50 = 1200 nM T53748 C8Y2RZ 44405311 IC50 = 190 nM T53748 C5OP2U 44405314 IC50 = 560 nM T53748 C6LV7J 44405327 IC50 = 550 nM T53748 C6TH2N 44405330 IC50 = 413 nM T53748 C37YBD 44405336 IC50 = 2500 nM T53748 C85YLH 44405338 IC50 = 140 nM T53748 C9K2TE 44405339 IC50 = 160 nM T53748 C6XVI1 44405380 IC50 = 320 nM T53748 C98SNV 44410066 IC50 = 22000 nM T53748 CB2G1Q 44410081 IC50 = 19000 nM T53748 C7DWG8 44410086 IC50 = 11000 nM T53748 C4MJ7O 44410094 IC50 = 7200 nM T53748 C4SV1O 44410097 IC50 = 28000 nM T53748 C3YI5T 44410098 IC50 = 27000 nM T53748 CU26VN 44410128 IC50 = 46000 nM T53748 CGP8A4 44410129 IC50 > 50000 nM T53748 CKAN96 44410130 IC50 = 3300 nM T53748 CL2V1B 44410133 IC50 = 18000 nM T53748 CZ38PQ 44410134 IC50 = 19000 nM T53748 C5RNT6 44410138 IC50 > 50000 nM T53748 C2K3EJ 44410170 IC50 = 15000 nM T53748 C26ODM 44410210 IC50 = 35000 nM T53748 C14ORH 44410211 IC50 > 50000 nM T53748 C3B0KG 44410215 IC50 > 50000 nM T53748 CL47JF 44410233 IC50 > 50000 nM T53748 CBVJ69 44410234 IC50 = 6100 nM T53748 CXDQ24 44410238 IC50 = 11000 nM T53748 CS50BT 44410252 IC50 > 50000 nM T53748 C1M4PV 44410256 IC50 = 7200 nM T53748 CIWT26 44410284 IC50 = 10000 nM T53748 C8RIW6 44410286 IC50 = 35000 nM T53748 CJ8H7A 44410287 IC50 = 2500 nM T53748 CSEQ42 44410291 IC50 = 26000 nM T53748 CH1U8G 44410295 IC50 > 50000 nM T53748 CITZ07 44423245 IC50 > 100000 nM T53748 CYC1F5 44423251 IC50 > 100000 nM T53748 CQN15Z 44423263 IC50 = 40000 nM T53748 C2CTI4 44423264 IC50 = 50000 nM T53748 C9PSC6 44423265 IC50 = 70000 nM T53748 CP92HW 44437887 IC50 = 40 ug.mL-1 T53748 CB0T1D 49797329 IC50 = 5 ug.mL-1 T53748 CXAP09 49799790 IC50 = 20 ug.mL-1 T53748 CYVB76 56835122 IC50 = 91130 nM T53748 CC5K9J 135993357 IC50 = 100000 nM T53748 D00RIX 5280443 IC50 = 50000 nM T53748 D00TWC 15942656 IC50 = 440 nM T53748 D01DTE 21272512 IC50 = 220 nM T53748 D01TGI 25023954 IC50 = 140 nM T53748 D03DND 25023959 IC50 = 210 nM T53748 D05VXX 25023960 IC50 = 480 nM T53748 D07YDN 5281654 IC50 = 5000 nM T53748 D08BMM 6312649 IC50 = 0.3 ug.mL-1 T53748 D08EME 25023967 IC50 = 190 nM T53748 D08FBM 16220128 IC50 = 76 nM T53748 D08KNJ 25023966 IC50 = 230 nM T53748 D09QZL 44405331 IC50 = 120 nM T53748 D0A1XH 25023962 IC50 = 290 nM T53748 D0A7US 25023963 IC50 = 120 nM T53748 D0A9HU 44410251 IC50 = 7000 nM T53748 D0C6IE 1123 IC50 > 100 ug.mL-1 T53748 D0EW3L 5281222 Ki = 14 nM T53748 D0FW2W 25023968 IC50 = 38 nM T53748 D0G3TK 5280863 IC50 = 20000 nM T53748 D0JL2T 5393152 IC50 = 10000 nM T53748 D0L0AZ 25023961 IC50 = 180 nM T53748 D0L7HD 25023969 IC50 = 71 nM T53748 D0LU2N 25023958 IC50 = 110 nM T53748 D0MF5Y 5281614 IC50 = 1000 nM T53748 D0NJ4H 5281670 IC50 = 5000 nM T53748 D0O9UI 22947105 IC50 = 200 nM T53748 D0QV8V 16220126 IC50 = 440 nM T53748 D0RB1V 6419835 Ki = 40 nM T53748 D0T3PW 5281672 IC50 = 400 nM T53748 D0U7MR 25023955 IC50 = 49 nM T53748 D0X4BJ 6852148 IC50 = 360 nM T53748 D0Z7FM 6852143 IC50 = 180 nM T32780 C10SQP 439353 IC50 = 1049000 nM T32780 CO1N3W 11710828 IC50 = 113000 nM T32780 CJ9I0G 12900878 IC50 = 1828000 nM T32780 CADH05 12900879 IC50 = 2831000 nM T32780 D07ONX 64689 IC50 > 30000000 nM T14558 D02INZ 2387 IC50 = 51 nM T14558 D05QMJ 5287596 Ki = 10 nM T14558 CIK93A 3348131 Ki = 88 nM T14558 C49IOZ 6857707 Ki = 2.8 nM T14558 C7JAG9 9853336 Ki = 18 nM T14558 C87SWZ 9872983 Ki = 0.6 nM T14558 CA9Z4S 9875345 Ki = 0.07 nM T14558 C9OHQ3 10051587 Ki = 84 nM T14558 CRUS92 10111743 IC50 = 190 nM T14558 C9US7W 10112313 IC50 = 120 nM T14558 CK7S4F 10139527 Ki = 155 nM T14558 CGN3R6 10271568 IC50 = 200 nM T14558 C1HVW5 10294248 IC50 = 73 nM T14558 CJ9K8M 10294609 IC50 = 210 nM T14558 C0T3CN 10296435 IC50 = 5 nM T14558 C84DGQ 10327019 Ki = 210 nM T14558 CC3Z8U 10412364 Ki = 93 nM T14558 CB4X5P 10417378 Ki = 0.4 nM T14558 C48IUK 10864508 Ki = 38 nM T14558 C30EGA 10885646 Ki = 470 nM T14558 C2MV8C 10886082 Ki = 19 nM T14558 C8NHR5 10984568 Ki = 41 nM T14558 C8L2WC 11005945 Ki = 20 nM T14558 CEG83K 11135464 Ki = 73 nM T14558 CJ8P0B 11262416 IC50 = 2200 nM T14558 CBDM51 11354224 IC50 = 2400 nM T14558 CFS7T8 11540675 Ki = 1.3 nM T14558 C19ARJ 15984063 Ki = 5.4 nM T14558 C80YJG 16007063 Ki = 2.5 nM T14558 C9WCA6 44314160 Ki = 340 nM T14558 CT4O2N 44314174 Ki = 6900 nM T14558 C5KIL1 44314175 Ki = 870 nM T14558 C3XY7T 44314176 Ki = 300 nM T14558 CFJS82 44314388 Ki = 7400 nM T14558 C8H3AQ 44314393 Ki = 11000 nM T14558 CS2B3L 44314462 Ki = 24000 nM T14558 CHQ6K3 44314463 Ki = 9800 nM T14558 C3NC4I 44314464 Ki = 9700 nM T14558 C9YZQ3 44314474 Ki = 80000 nM T14558 CC25DH 44314493 Ki = 12000 nM T14558 C84GZN 44314494 Ki = 11000 nM T14558 C0MFA4 44314495 Ki = 29000 nM T14558 CP46GK 44314665 Ki = 50000 nM T14558 CW0XV9 44314666 Ki = 160 nM T14558 C7J5WH 44314667 Ki = 400 nM T14558 C02EFV 44314678 Ki = 7000 nM T14558 CQ3K9H 44314679 Ki = 6900 nM T14558 C6TU0R 44314680 Ki = 890 nM T14558 C2JWR0 44314690 Ki = 1300 nM T14558 C9J3YE 44314694 Ki = 13000 nM T14558 CZK42J 44314709 Ki = 16000 nM T14558 CEM7G4 44314742 Ki = 2600 nM T14558 C8AX1U 44314743 Ki = 370000 nM T14558 C9I6FR 44315066 Ki = 7300 nM T14558 CK61RF 44315079 Ki = 42000 nM T14558 CIBE78 44315607 Ki = 3 nM T14558 CZ3CY0 44315608 Ki = 5 nM T14558 C07NBY 44315609 Ki = 2000 nM T14558 C8DQ5R 44315610 Ki = 680 nM T14558 C71UBD 44315637 Ki = 150 nM T14558 C5QUO9 44315743 Ki = 100 nM T14558 CA8L4R 44315744 Ki = 15000 nM T14558 CPV7S5 44315758 Ki = 2 nM T14558 CZ8RS4 44315843 Ki = 90 nM T14558 CUGF09 44315844 Ki = 10 nM T14558 CX20QR 44315845 Ki = 101000 nM T14558 C4KF3H 44315846 Ki = 40 nM T14558 C0IVD5 44315849 Ki = 9 nM T14558 CAJ97K 44316048 Ki = 366 nM T14558 CQ52SH 44316049 Ki = 31 nM T14558 C1MRI0 44316050 Ki = 5 nM T14558 CSY03Q 44350110 Ki = 33 nM T14558 CN5H9Q 44350175 Ki = 250 nM T14558 C87NXA 44350193 Ki = 90 nM T14558 C4Y3TQ 44350195 Ki = 180 nM T14558 C0Q7KU 44350214 IC50 = 2 nM T14558 CP5Z3F 44350231 Ki = 330 nM T14558 C7VTQ8 44385971 Ki = 350 nM T14558 C4MY8T 44386061 Ki = 10 nM T14558 CW73FL 44386111 Ki = 180 nM T14558 CDV0B1 44386147 Ki = 13700 nM T14558 CHK5A4 44386595 Ki = 2400 nM T14558 CKP6V3 44386640 Ki = 213000 nM T14558 C6FDC2 44390015 IC50 = 4400 nM T14558 C6BQ8N 44390025 IC50 = 19900 nM T14558 CHD59A 44390036 IC50 = 23600 nM T14558 CV5RX2 44390046 IC50 = 12800 nM T14558 CB0C2E 44390058 IC50 = 21300 nM T14558 C5RNL7 44390059 IC50 = 9090 nM T14558 C46JUY 44390060 IC50 = 12400 nM T14558 CVM2Y5 44390082 IC50 = 4700 nM T14558 C8V0CX 44390106 IC50 = 9300 nM T14558 C2R0NL 44390107 IC50 = 5700 nM T14558 CO8J3W 44390109 IC50 = 4100 nM T14558 COBM92 44390218 IC50 = 5900 nM T14558 CNQS07 44394012 Ki = 290 nM T14558 CV6O7K 44394163 Ki = 970 nM T14558 CC0V8I 44394165 Ki = 1238 nM T14558 CH58JG 44394177 Ki = 1550 nM T14558 C90IZA 44394186 Ki = 875 nM T14558 CO2XU5 44394199 Ki = 518 nM T14558 C16QXM 44394232 Ki = 1550 nM T14558 C6AUQ8 44394236 Ki = 580 nM T14558 CD7U5E 44394267 Ki = 615 nM T14558 C8QPS0 44394278 Ki = 426 nM T14558 CBU59Y 44394342 Ki = 390 nM T14558 CPNZ96 44394575 Ki = 245 nM T14558 CVK4W3 44394662 Ki = 138 nM T14558 CY09ES 44396504 Ki = 1.5 nM T14558 C4X2OS 44396541 Ki = 88 nM T14558 CY80RP 44396542 Ki = 4.3 nM T14558 C6JK2D 44396602 Ki = 59 nM T14558 C32ATR 44398672 Ki = 240 nM T14558 CO8R6N 44398687 Ki = 101 nM T14558 CN84TJ 44398709 Ki > 20000 nM T14558 C81XZC 44398838 Ki = 373 nM T14558 C1XY3O 44398882 Ki = 197 nM T14558 C7RDV3 44398890 Ki > 20000 nM T14558 C1U4YR 44398931 Ki = 61 nM T14558 C8G4XK 44398933 Ki = 368 nM T14558 C4XFB1 44399237 Ki = 290 nM T14558 CXEJ41 44399289 Ki = 310 nM T14558 CMT9K2 44399296 Ki = 41 nM T14558 CB7GU1 44399302 Ki = 125 nM T14558 CU04PG 44399314 Ki = 141 nM T14558 CAZC79 44399329 Ki = 41 nM T14558 CAM61E 44399337 Ki = 57 nM T14558 CQ96KT 44399350 Ki = 116 nM T14558 CDB3U2 44399365 Ki = 32 nM T14558 C01ILA 44399375 Ki = 68 nM T14558 CO91RY 44399384 Ki = 246 nM T14558 CCJY60 44399416 Ki = 497 nM T14558 C9XGC4 44399419 Ki = 49 nM T14558 C9RHE1 44399426 Ki = 124 nM T14558 C1UCS5 44399506 Ki = 185 nM T14558 CY2KB9 44399512 Ki = 162 nM T14558 C2A1GS 44399522 Ki = 128 nM T14558 C4E7BY 44411566 IC50 = 1600 nM T14558 CKEM18 44411580 IC50 = 130 nM T14558 CG3KB9 44411617 IC50 = 5100 nM T14558 CQK14J 44411620 IC50 = 5600 nM T14558 CO5BF2 44411621 IC50 = 5700 nM T14558 CQD1P3 44411626 IC50 = 760 nM T14558 CN8GR3 44411792 IC50 = 1300 nM T14558 C3YL4G 44411807 IC50 = 270 nM T14558 C29ULX 44411828 IC50 = 810 nM T14558 CC5Y7F 44411942 IC50 = 21100 nM T14558 CB1G3D 44412151 Ki = 6200 nM T14558 CC2Z1K 44412258 Ki = 2500 nM T14558 CLQ54S 44412280 Ki = 30000 nM T14558 C78DIR 44412515 Ki = 46 nM T14558 CY0LK9 44412517 Ki = 5 nM T14558 CUOX14 44412519 Ki = 32 nM T14558 C7L0RD 44412532 Ki = 5 nM T14558 C61QCJ 44412534 Ki = 9.6 nM T14558 CLU6F4 44412546 Ki = 2.9 nM T14558 C4TYG5 44412554 Ki = 11 nM T14558 C57SNK 44412556 Ki = 6.55 nM T14558 C18TWV 44412563 Ki = 4.7 nM T14558 C5ST8F 44412580 Ki = 18 nM T14558 C9WPJ4 44412584 Ki = 4.6 nM T14558 CWG5V4 44412591 Ki = 9.2 nM T14558 CKR4O6 44412601 Ki = 6.8 nM T14558 CGH3S6 44412610 Ki = 5.7 nM T14558 C8OE5N 44412615 Ki = 6.2 nM T14558 CBOJ83 44412620 Ki = 9.8 nM T14558 C3AU5P 44412629 Ki = 5.8 nM T14558 CWF72Q 44412631 Ki = 3.25 nM T14558 CUG10P 44412693 Ki = 17 nM T14558 CD7VO3 44412744 Ki = 2.3 nM T14558 C8LA7C 44412763 Ki = 6.5 nM T14558 C3BX5Y 44412781 Ki = 7.6 nM T14558 CS8DA4 44412785 Ki = 22 nM T14558 CA5G2R 44412795 Ki = 3.75 nM T14558 CJF45Q 44412803 Ki = 3.7 nM T14558 C5Q7LD 44413973 Ki = 10 nM T14558 CI4BX0 44413974 Ki = 96 nM T14558 CBP63U 44414061 Ki = 24 nM T14558 C0HMI7 44414062 Ki = 78 nM T14558 CR2I5B 44414080 Ki = 27 nM T14558 C54RLJ 44414103 Ki = 19 nM T14558 COTK13 44414104 Ki = 41 nM T14558 CH73SZ 44414147 Ki = 1100 nM T14558 C1SP4A 44414165 Ki = 13 nM T14558 CWUI89 44414193 Ki = 25 nM T14558 CMS23E 44414210 Ki = 360 nM T14558 C85UJB 44414227 Ki = 120 nM T14558 C08MJX 44414236 Ki = 2700 nM T14558 CS8B0C 44414252 Ki = 180 nM T14558 C5NZ2H 44414259 Ki = 16 nM T14558 C8JL0A 44414268 Ki = 12 nM T14558 CV52XQ 44414273 Ki = 14 nM T14558 CMR30P 44414330 Ki = 16 nM T14558 CR6B8L 44414331 Ki = 1.8 nM T14558 CBAT52 44414332 Ki = 2.9 nM T14558 CO8A0Y 44414333 Ki = 3.7 nM T14558 C9B1RY 44414334 Ki = 1.8 nM T14558 CU7XR2 44414335 Ki = 1.7 nM T14558 C6FTY7 44414336 Ki = 1.7 nM T14558 CP3H4U 44414341 Ki = 1.9 nM T14558 C75KJO 44414360 Ki = 1.5 nM T14558 CL19PK 44414361 Ki = 1.9 nM T14558 C2WK3C 44414362 Ki = 2.1 nM T14558 C7N6RE 44414406 Ki = 3 nM T14558 C07IFH 44414407 Ki = 60 nM T14558 CAJ0B9 44414408 Ki = 140 nM T14558 CQU27H 44414409 Ki = 3.6 nM T14558 C0NQL2 44414410 Ki = 220 nM T14558 CJN0G9 44414411 Ki = 8.2 nM T14558 C81XCL 44414412 Ki = 3.5 nM T14558 CCU57L 44414430 Ki = 39 nM T14558 CSX2D1 44414431 Ki = 11 nM T14558 CY1MW2 44414438 Ki = 2.4 nM T14558 CV3N1P 44414454 Ki = 9.9 nM T14558 C7PZ6S 44414474 Ki = 11 nM T14558 C9C4XJ 44414482 Ki = 2 nM T14558 CFLR38 44414489 Ki = 5.8 nM T14558 CF5L6K 44414510 Ki = 770 nM T14558 CTG1N5 44414511 Ki = 37 nM T14558 C8I2QP 44414559 Ki = 34 nM T14558 C1JXO7 44414560 Ki = 470 nM T14558 C1NOI8 44414566 Ki = 13 nM T14558 C8QD3M 44414567 Ki = 3.2 nM T14558 CSTD86 44414582 Ki = 230 nM T14558 CN19RU 45261811 Ki = 140 nM T14558 CJ5E2P 45265199 Ki = 22 nM T14558 C78DJQ 71711730 IC50 < 10000 nM T14558 D09OBJ 9872263 Ki = 6.5 nM T14558 D0Y5IQ 44255320 IC50 = 10000 nM T94197 D03ZBT 11626560 IC50 > 10000 nM T94197 D0B5LF 448042 IC50 = 600 nM T94197 D03KKR 3547 IC50 = 780 nM T94197 D03LWG 53235510 IC50 > 10000 nM T94197 D07EHV 44814409 IC50 > 10000 nM T94197 D0E3TC 44259 IC50 = 1.97 nM T94197 D03BNU 59604787 IC50 > 10000 nM T94197 C9O3XQ 9901617 IC50 = 70 nM T94197 CU0E8O 11690457 Ki = 77 nM T94197 C9TU1O 16046126 IC50 > 1000 nM T94197 CK60ZM 24758992 IC50 = 2300 nM T94197 CZ2PQ6 24863113 IC50 = 110 nM T94197 CBYM61 24863535 IC50 = 1400 nM T94197 CY8L7E 24896769 IC50 > 10000 nM T94197 C1ONA4 24996161 IC50 = 17 nM T94197 CZO27W 25054032 IC50 > 5000 nM T94197 CN2G3K 25054307 IC50 > 5000 nM T94197 C7IZ6K 25055317 IC50 > 5000 nM T94197 CFHO90 25056112 IC50 = 1600 nM T94197 CU8X0H 25056370 IC50 = 1700 nM T94197 CV15HY 25056371 IC50 > 5000 nM T94197 C76LFY 25056889 IC50 > 5000 nM T94197 CH6AU8 25057408 IC50 = 4400 nM T94197 C0B7RT 25057409 IC50 > 5000 nM T94197 C3AT0H 25057667 IC50 > 5000 nM T94197 CH7YC4 25057933 IC50 > 5000 nM T94197 CSI0U1 44819541 IC50 = 770 nM T94197 CLS29B 46872626 IC50 > 10000 nM T94197 CXUO70 46890036 IC50 = 510 nM T94197 CZ2V8R 46890138 IC50 = 3000 nM T94197 CSV5B9 46901859 IC50 = 7 nM T94197 CEQN27 52936621 Ki > 1000 nM T94197 C2W9OA 53324451 IC50 > 10000 nM T94197 C1XS2J 54760383 IC50 > 10000 nM T94197 C1MR8Q 60097495 IC50 > 10000 nM T94197 C1HSE0 67035086 IC50 = 2400 nM T94197 CWI6K5 67035106 IC50 > 10000 nM T94197 CV63UL 67240318 IC50 > 10000 nM T94197 CD56XK 68293660 IC50 > 10000 nM T94197 CSV23A 78673872 IC50 = 742 nM T94197 CPG3A5 86302574 IC50 > 30000 nM T94197 CN67RP 91758287 IC50 = 974 nM T94197 C7ZL3Q 118715599 IC50 = 58 nM T94197 C8T0AY 118715600 IC50 = 995 nM T94197 C2J3YZ 118715601 IC50 = 920 nM T94197 CRG06J 118715602 IC50 = 951 nM T94197 C7WS3V 118715603 IC50 > 1000 nM T94197 CQM81J 118715604 IC50 > 1000 nM T94197 C2MD1Q 155513187 IC50 > 10000 nM T94197 D00ERW 44444843 Ki > 8195 nM T94197 D06HVH 54613583 IC50 = 300 nM T94197 D0N1UU 46871820 IC50 = 14 nM T94197 D0V0KA 24863112 IC50 > 8000 nM T20575 D00XBC 46861584 IC50 > 10000 nM T20575 C7Y8VS 1318 EC50 = 3900 nM T20575 CB4Z9P 1474 EC50 = 39810.72 nM T20575 C78GSK 14338 EC50 = 3162.28 nM T20575 CW6J7R 15664 EC50 = 7500 nM T20575 CBX47E 20445 EC50 = 4800 nM T20575 CD72TB 65237 EC50 < 1000000 nM T20575 CF1UA4 70848 EC50 = 4900 nM T20575 CR15FN 72791 EC50 = 1995.26 nM T20575 C8SC9N 72792 EC50 = 501.19 nM T20575 C7SIE4 74265 EC50 = 480 nM T20575 CMJ4V7 77524 EC50 = 79432.82 nM T20575 CGZ1C6 77865 EC50 = 3000 nM T20575 CBW4N5 93149 EC50 = 630.96 nM T20575 CTUE81 336912 EC50 < 1000000 nM T20575 C2P3FM 353741 EC50 < 1000000 nM T20575 CSF9D4 602123 EC50 < 1000000 nM T20575 CXMY27 619353 EC50 < 1000000 nM T20575 CYU56N 667748 EC50 = 390 nM T20575 C4WCL7 792361 Ki = 2600 nM T20575 C8EA0N 1099153 Ki = 7745 nM T20575 CAF8P7 2733927 EC50 = 5011.87 nM T20575 C2PZ0U 3384970 Ki = 42.6 nM T20575 C9P4WR 3594744 Ki > 30000 nM T20575 CYVR59 3989497 Ki > 30000 nM T20575 CMV9K7 5335896 Ki > 44000 nM T20575 C54BLX 9911916 IC50 = 25.12 nM T20575 C13UYJ 9982672 Ki = 2.3 nM T20575 C6WOU1 9984180 Ki = 1.1 nM T20575 CUQF40 10003657 IC50 = 39.81 nM T20575 C6XCG1 10004785 IC50 = 1258.93 nM T20575 C24SKQ 10006907 Ki = 0.7 nM T20575 C9VN0R 10254576 Ki = 4.1 nM T20575 C9FA0W 10255258 IC50 = 50.12 nM T20575 CWFB30 10323427 IC50 > 1000 nM T20575 CL2Z9Q 10343818 IC50 = 630.96 nM T20575 C3GOJ4 10367938 Ki = 0.17 nM T20575 C5GDY0 10391001 Ki = 0.3 nM T20575 CU0Y3K 10391077 Ki = 5.21 nM T20575 CXH36J 10409369 IC50 = 501.19 nM T20575 C4LXQ0 10412437 IC50 = 3162.28 nM T20575 CSBN34 10412573 IC50 = 794.33 nM T20575 CA3MG8 10433657 IC50 = 251.19 nM T20575 CS9WA0 10479253 IC50 = 31.62 nM T20575 C0G5HP 10480554 IC50 = 125.89 nM T20575 CZJA18 11212011 Ki > 30000 nM T20575 CUH4F5 11235229 Ki = 578 nM T20575 CK36XS 11273324 IC50 = 81.28 nM T20575 C1RB4T 11329260 Ki = 9.5 nM T20575 C9NG0M 11384528 Ki = 3277 nM T20575 CYLF54 11452569 Ki = 4.4 nM T20575 C6ZN1O 11502217 Ki = 1400 nM T20575 C0QK6P 11519336 Ki = 11 nM T20575 CMC5B1 11526626 Ki = 15 nM T20575 CRJC25 11530171 Ki = 9100 nM T20575 CFU5V9 11533398 IC50 = 11 nM T20575 CQZ82F 11539239 IC50 = 55 nM T20575 CVX6L8 11541073 Ki = 250 nM T20575 C8P5GF 11541506 IC50 = 1 nM T20575 C7B4YX 11563243 Ki = 23 nM T20575 CXJ8W9 11584004 IC50 = 22 nM T20575 C6M4TY 11681610 Ki = 9200 nM T20575 CRF5P4 11685733 IC50 = 4 nM T20575 C04VLB 11706579 Ki = 60 nM T20575 C0TU4A 11754900 Ki = 0.7 nM T20575 CD0F5T 11842667 IC50 = 26.92 nM T20575 CQSU51 11950826 IC50 = 165.96 nM T20575 C85VJZ 11950827 IC50 = 79.43 nM T20575 CQVX45 11950828 IC50 = 114.82 nM T20575 C0WVX4 11951000 IC50 = 33.11 nM T20575 C8SZH2 11965686 IC50 = 54.95 nM T20575 CK80NA 12987698 EC50 = 6309.57 nM T20575 CJGC50 14434082 EC50 = 15000 nM T20575 CIZ8C1 15783796 EC50 = 630.96 nM T20575 CEZI54 16064872 IC50 = 2.63 nM T20575 C96FEP 16065425 IC50 = 128.82 nM T20575 CVCJ16 16065428 IC50 = 1479.11 nM T20575 C6MC0Z 16065567 IC50 = 30.9 nM T20575 CPN9H5 16065569 IC50 = 8.128 nM T20575 CL1M3W 16065704 IC50 = 6.607 nM T20575 C2Y0BN 16105759 Ki > 44000 nM T20575 CR8HI6 16105760 Ki = 15.2 nM T20575 CY9SB1 16105765 IC50 > 3300 nM T20575 COK21G 16105771 IC50 = 9.5 nM T20575 CL4E0W 16105772 IC50 = 19.2 nM T20575 C3B2ZP 16105773 IC50 = 59.5 nM T20575 C7L6WA 16105774 IC50 = 15.3 nM T20575 CA32CK 16105775 IC50 = 36.1 nM T20575 CUK8W2 16105776 IC50 = 24.6 nM T20575 CRC6L3 16105777 IC50 = 23.6 nM T20575 C8I5WV 16105778 IC50 = 46.9 nM T20575 C3SX2F 16105779 IC50 = 43.9 nM T20575 C8JOX2 16105780 IC50 = 1004 nM T20575 CHJ5T0 16105781 IC50 = 41.7 nM T20575 C4NY7S 16105782 IC50 = 100 nM T20575 CQ5B8S 16105783 IC50 = 57.9 nM T20575 CD7M2B 16105784 IC50 = 6.1 nM T20575 CZ1J9M 16105785 IC50 > 1900 nM T20575 CPK35J 16105786 IC50 = 638.5 nM T20575 CUMD39 16105787 IC50 = 612.5 nM T20575 CX5KI3 16105788 Ki = 1.6 nM T20575 CQ8R1J 16105798 Ki > 5000 nM T20575 CZ87JP 16105799 Ki = 16.4 nM T20575 C3ENO5 16105802 Ki = 2.5 nM T20575 CKXP12 16105803 Ki = 6.7 nM T20575 CK28NO 16105804 Ki = 9.1 nM T20575 C7IW2N 16105805 Ki = 15.8 nM T20575 CO19JS 16105807 Ki = 11.3 nM T20575 CVO9B7 16105809 Ki = 199 nM T20575 CHX6F7 16105811 Ki = 1.5 nM T20575 C81BMQ 16105813 Ki = 114 nM T20575 CE9R1V 16105815 IC50 = 9.8 nM T20575 C5E2DX 16105817 IC50 = 4.2 nM T20575 C64DZP 16105819 IC50 = 19.6 nM T20575 C1HZ9D 16105820 Ki = 77.4 nM T20575 C2S3AQ 16105821 Ki = 77.7 nM T20575 C8J5WR 16105822 Ki = 1.6 nM T20575 CP3YM1 16105824 Ki = 4.2 nM T20575 CFLK94 16105826 Ki = 71 nM T20575 CP9Q7T 16105830 Ki = 566.5 nM T20575 C9VKP4 16105831 Ki = 125.6 nM T20575 CH2F6A 16105832 Ki = 34.3 nM T20575 C6UN3Q 16105834 Ki > 15000 nM T20575 C0I3AL 16105836 IC50 > 3300 nM T20575 C78VEF 16105840 Ki = 37.9 nM T20575 CB9HM4 16105843 Ki > 5000 nM T20575 C27NRT 16105844 Ki = 50.9 nM T20575 C4VW7B 16105847 Ki > 30000 nM T20575 CKBO86 16105854 IC50 = 144.5 nM T20575 CVU10F 16105855 IC50 = 205.9 nM T20575 C7PJI0 16105856 IC50 = 7.65 nM T20575 CBA38K 16105857 IC50 = 12.5 nM T20575 CFK1O9 16105858 IC50 = 5.1 nM T20575 C1CZF3 16105859 IC50 = 20 nM T20575 C3MZO5 16105860 IC50 = 10.8 nM T20575 CW25VQ 16105861 IC50 = 6.9 nM T20575 C85YRI 16105862 IC50 = 1519 nM T20575 CIH0N4 16105863 IC50 = 37 nM T20575 CEGN62 16105864 IC50 = 20.4 nM T20575 CF4LC0 16105865 IC50 = 280 nM T20575 CU8O9M 16105866 IC50 = 885.1 nM T20575 C56LRM 16105867 IC50 = 367.7 nM T20575 CU06LQ 16105868 IC50 = 365 nM T20575 CYTD60 16105876 Ki = 7.2 nM T20575 C28HEZ 16105877 Ki = 5.4 nM T20575 CRSY15 16105880 Ki = 1.6 nM T20575 CJCG76 16105882 Ki = 81.1 nM T20575 C2IZK6 16105885 IC50 = 14.5 nM T20575 CK94HY 16105887 IC50 = 28.6 nM T20575 CG9X0C 16105888 Ki = 243 nM T20575 C1SW7R 16105889 Ki = 2.2 nM T20575 C24BPX 16105890 Ki = 108 nM T20575 CA9XR0 16105891 Ki = 3.5 nM T20575 CP5B9N 16105892 Ki = 4.2 nM T20575 C0RF4V 16105893 Ki = 6.3 nM T20575 CI4E3G 16105895 Ki = 2033 nM T20575 CKPQ93 16112836 IC50 = 19.95 nM T20575 CM0V6H 44419031 Ki = 45.6 nM T20575 CVA73W 44419032 Ki = 35.7 nM T20575 CKA7Z0 44419035 Ki = 32.1 nM T20575 CXG9O0 44419086 Ki > 44000 nM T20575 C0SQ3G 44439837 IC50 = 1584.89 nM T20575 CV6I5H 44439838 IC50 = 6309.57 nM T20575 CYV10A 44439839 IC50 < 50118.72 nM T20575 CEA1I5 44439840 IC50 < 50118.72 nM T20575 CV4N3Z 44439841 IC50 < 50118.72 nM T20575 CUVO37 44439842 IC50 < 50118.72 nM T20575 CMO70Y 44439843 IC50 = 1000 nM T20575 CCR1Z6 44439844 IC50 < 50118.72 nM T20575 CTJB51 44439845 IC50 < 50118.72 nM T20575 C59BFI 44439846 IC50 < 50118.72 nM T20575 CFU53W 44439864 IC50 < 50118.72 nM T20575 C2ESO7 44439865 IC50 < 50118.72 nM T20575 C9N5AS 44439881 IC50 = 1258.93 nM T20575 CV0DH4 44439883 IC50 = 3162.28 nM T20575 C63YBE 44439884 IC50 < 50118.72 nM T20575 CRL70X 44439885 IC50 = 7943.28 nM T20575 C8RV9U 44439886 IC50 = 12589.25 nM T20575 CV75QH 44439887 IC50 = 6309.57 nM T20575 CXMR49 44439888 IC50 < 50118.72 nM T20575 C8SPT1 44439890 IC50 = 1258.93 nM T20575 C1NMR0 44439895 IC50 = 12589.25 nM T20575 C7E0YR 44439900 IC50 < 50118.72 nM T20575 CCD86W 44439909 IC50 = 6309.57 nM T20575 CFS76J 44439911 IC50 < 50118.72 nM T20575 CVA46I 44456948 IC50 = 27.54 nM T20575 CI71FO 44456993 IC50 = 18.2 nM T20575 CT5H0R 44457009 IC50 = 12.02 nM T20575 CTCQ07 44457046 IC50 = 19.05 nM T20575 CRSI16 44457089 IC50 = 16.22 nM T20575 C2XZN7 44457090 IC50 = 11.48 nM T20575 CE6U0F 44457093 IC50 = 33.11 nM T20575 CPK1J7 44457105 IC50 = 34.67 nM T20575 CF4YN8 44598057 IC50 = 107.15 nM T20575 C9MT0V 44598058 IC50 = 4.898 nM T20575 C71QNY 44598059 IC50 = 141.25 nM T20575 C9TH0G 44598060 IC50 = 1819.7 nM T20575 CZWY54 44598061 IC50 = 95.5 nM T20575 CP27OH 44598062 IC50 = 5.623 nM T20575 CS76XZ 44598121 IC50 = 22.39 nM T20575 C0L4FZ 44598124 IC50 = 2.63 nM T20575 CGQT32 44598769 IC50 = 141.25 nM T20575 CG2SD8 44598819 IC50 = 70.79 nM T20575 C27GZB 44598820 IC50 = 524.81 nM T20575 CV9G1H 44598821 IC50 = 14.79 nM T20575 CE4LA5 45483880 IC50 = 2.818 nM T20575 CX12QY 45483901 IC50 = 2.399 nM T20575 C0TED2 45483913 IC50 = 22.39 nM T20575 C6ENV5 100951623 EC50 > 10000 nM T20575 CADQ93 155557362 IC50 = 5200 nM T20575 D0K8BZ 11774008 Ki = 1760 nM T20575 D0M1AE 11270007 Ki = 233.1 nM T56175 D0I2YV 501398 IC50 = 1150 nM T56175 D0X3GG 1949 IC50 = 223.87 nM T56175 CE3XT6 445986 IC50 = 16 nM T56175 CG2SH5 445987 IC50 = 19.05 nM T56175 CMZ90J 445988 IC50 = 6.457 nM T56175 C4IFB0 445989 IC50 = 19.5 nM T56175 C0D9BA 445990 IC50 = 29 nM T56175 C90LVU 445991 IC50 = 1905.46 nM T56175 CW3X0J 445992 IC50 = 2.884 nM T56175 C05YIN 447553 IC50 = 3.5 nM T56175 C65XKW 447559 IC50 = 500 nM T56175 C01LPN 447560 IC50 = 616.6 nM T56175 C0K5CF 447562 IC50 = 11.3 nM T56175 C70PUX 501376 IC50 = 92 nM T56175 C7T3AD 748374 IC50 = 4750 nM T56175 CZ1S6P 6438755 IC50 = 3000 nM T56175 CO28YI 6479040 IC50 = 4.3 nM T56175 C8FTY4 7995534 IC50 = 1380 nM T56175 CGME20 8851244 IC50 = 1410 nM T56175 C8VD2O 8851269 IC50 = 12700 nM T56175 CP9HS7 9114889 IC50 = 3120 nM T56175 CR52CZ 9535392 IC50 = 10800 nM T56175 CN73CV 9870902 IC50 = 112 nM T56175 C8GSR0 9890308 IC50 = 640 nM T56175 C4NU1E 9952802 IC50 = 3 nM T56175 CGH6M2 9959583 IC50 = 5.7 nM T56175 C0PT7L 10138152 IC50 = 5 nM T56175 C32QWP 10159157 IC50 = 10 nM T56175 CUCG94 10160616 IC50 = 230 nM T56175 CGC42D 10297203 IC50 = 11500 nM T56175 C8CD5R 10502890 IC50 = 8400 nM T56175 C46KCR 10577130 IC50 = 37 nM T56175 CS1YQ2 10665993 IC50 = 15000 nM T56175 CKG16M 10693131 IC50 = 143 nM T56175 C4U6RL 10743771 IC50 = 161 nM T56175 C46BFN 10765813 IC50 = 540 nM T56175 CE2U3Y 10862930 IC50 = 8.7 nM T56175 C1TCE8 10885481 IC50 = 7.8 nM T56175 CA5UH1 10917490 IC50 = 5.6 nM T56175 CZ1TJ9 10928636 IC50 = 4.571 nM T56175 CVT70N 10981049 IC50 = 22.39 nM T56175 C96SGO 10994090 IC50 = 12.3 nM T56175 C0PH6M 11003804 IC50 = 1.9 nM T56175 CA1GC9 11014097 IC50 = 6.7 nM T56175 COJ6D2 11015786 IC50 = 15.7 nM T56175 C4HB0V 11048762 IC50 = 4.074 nM T56175 C7E2SF 11059310 IC50 = 31.62 nM T56175 C10XTN 11091286 IC50 = 5.37 nM T56175 C9GY4R 11102507 IC50 = 11.4 nM T56175 CSJ3Z2 11113277 IC50 = 4.074 nM T56175 CX80TM 11123614 IC50 = 6.166 nM T56175 C2GW3J 11144462 IC50 = 35.3 nM T56175 CR1C6T 11144768 IC50 = 6.3 nM T56175 C7EL9N 11475734 IC50 = 28.7 nM T56175 C8C0KD 11729939 IC50 = 380 nM T56175 CFOZ08 11730147 IC50 = 7.9 nM T56175 C3CL7R 11743563 IC50 = 2.3 nM T56175 CG9TD0 15000175 IC50 > 100000 nM T56175 CAS74N 16655050 IC50 = 1100 nM T56175 CY0ZW7 18434247 IC50 = 97.72 nM T56175 C64UBJ 22313933 IC50 = 120 nM T56175 C2X4KN 22314073 IC50 = 4600 nM T56175 CO6JI1 22567752 IC50 = 2440 nM T56175 CUV39Q 22567773 IC50 = 100 nM T56175 C04LJY 22567802 IC50 = 450 nM T56175 CEYR19 22567883 IC50 = 440 nM T56175 CTS6N3 22567916 IC50 = 4930 nM T56175 CC9JK6 22568056 IC50 = 720 nM T56175 CZ0E4H 25022620 IC50 = 32 nM T56175 C59UCE 25022621 IC50 = 32 nM T56175 C0YP5N 44275335 IC50 = 430 nM T56175 CS6GQ2 44275353 Ki = 110 nM T56175 CJU1Y6 44306060 IC50 = 28.84 nM T56175 CKD6Y8 44306062 IC50 = 70.79 nM T56175 C0ROJ7 44306071 IC50 = 38.9 nM T56175 CO2L4P 44306091 IC50 = 1862.09 nM T56175 C3DCL5 44306371 IC50 = 47.86 nM T56175 CQ2EB4 44306372 IC50 = 240 nM T56175 CQ4C5G 44306432 IC50 = 13.49 nM T56175 CQU4J3 44306452 IC50 = 21.88 nM T56175 C7LHQ3 44306453 IC50 = 436.52 nM T56175 C45DPA 44341640 IC50 = 5.4 nM T56175 CUH4G9 44341779 IC50 = 4.1 nM T56175 CSB43N 44341780 IC50 = 20340 nM T56175 CC2R1M 44341784 IC50 = 19.6 nM T56175 C3RL1V 44341981 IC50 = 2.9 nM T56175 C9L4IN 44368021 IC50 = 1500 nM T56175 CF02EG 44368022 IC50 > 100000 nM T56175 CFSD76 44368023 IC50 = 70000 nM T56175 C9PCZ3 44368035 IC50 = 18000 nM T56175 CT6J7P 44368036 IC50 = 1000 nM T56175 CV3ER5 44368070 IC50 = 5000 nM T56175 CUI71Y 44427924 IC50 = 7.762 nM T56175 CB2ND4 44427932 IC50 = 19.05 nM T56175 CC90EF 44427946 IC50 = 19.5 nM T56175 C1XGI2 44440594 IC50 = 4500 nM T56175 CT0GH4 44440595 IC50 = 850 nM T56175 C4G6XK 44570900 IC50 = 270 nM T56175 CRW82M 44570901 IC50 = 90000 nM T56175 CDY2S0 44570982 IC50 = 100 nM T56175 CQX4Y1 44571035 IC50 > 1000 nM T56175 C30XZL 44571037 IC50 = 4120 nM T56175 C1G3EN 44571108 IC50 > 10000 nM T56175 CZVA80 44586247 EC50 = 100 nM T56175 C9P7FA 44586249 IC50 = 28 nM T56175 CL84KP 44586250 IC50 = 63 nM T56175 C7S3UF 44586287 IC50 = 500 nM T56175 C6AFB4 44586288 IC50 = 13 nM T56175 C1B0LZ 44586289 IC50 = 3 nM T56175 CT23XY 44586290 IC50 = 316 nM T56175 CY3QT0 44586291 IC50 = 2511 nM T56175 CV40KW 44586331 IC50 = 40 nM T56175 C6OPU4 44586332 IC50 = 20 nM T56175 C8AV1M 44586333 IC50 = 6 nM T56175 C7T0WE 45261590 IC50 = 3.5 nM T56175 CV84OH 46946069 IC50 = 35400 nM T56175 C4VM1K 46946070 IC50 = 58800 nM T56175 CO4S5W 56834930 IC50 = 5020 nM T56175 C8XN7W 60154274 IC50 = 7.8 nM T56175 C5PBR1 71456888 IC50 = 11.2 nM T56175 CEFO07 72199012 IC50 = 1000 nM T56175 CI1S2D 72199013 IC50 > 20000 nM T56175 C8MTH0 72199014 IC50 = 4500 nM T56175 CO1KS6 72199015 IC50 = 11900 nM T56175 CHMB42 72199016 IC50 = 12500 nM T56175 CXN2L8 72199018 IC50 > 20000 nM T56175 CI5EO6 127041210 IC50 = 2060 nM T56175 CS6D0W 127041211 IC50 = 2060 nM T56175 CI4J8Y 127041213 IC50 = 8510 nM T56175 CZ57EU 127041496 IC50 = 2510 nM T56175 CV9T0L 127041498 IC50 = 5280 nM T56175 CG7RY8 127041500 IC50 > 10000 nM T56175 CS6L4R 127042121 IC50 = 4220 nM T56175 CD2U9H 127042122 IC50 = 510 nM T56175 CT1U7D 145966025 IC50 = 120 nM T56175 CX16LD 145966143 IC50 = 230 nM T56175 CK3RJ1 145977714 IC50 = 16 nM T56175 D00XPB 44570860 IC50 = 250 nM T56175 D00ZEY 22314173 IC50 = 260 nM T56175 D0C7PY 15433 IC50 = 2150 nM T56175 D0K3TQ 10095126 IC50 = 0.22 nM T56175 D0R1EO 501375 IC50 = 16000 nM T56175 D0Z3CK 10138707 IC50 = 17.8 nM T82146 D02DGU 444795 Ki = 0.04 nM T82146 D0BM5G 5381 EC50 = 40 nM T82146 D0G3PI 449171 Ki = 1 nM T82146 D0JC9N 60164 EC50 = 3.1 nM T82146 D0K5ER 5281055 Ki = 10000 nM T82146 D0N0RU 82146 Ki = 130 nM T82146 D02GTY 108143 EC50 = 591 nM T82146 D06FOU 11518241 EC50 = 7.7 nM T82146 D06QXI 9863342 EC50 = 200 nM T82146 D08JAC 5288209 Ki > 400 nM T82146 D09YFJ 135411 EC50 = 49 nM T82146 D08GRF 5287705 EC50 = 0.34 nM T82146 D0YO4D 3922 Ki = 9901 nM T82146 C7QAB1 2418 EC50 = 51 nM T82146 CZBJ59 119342 Ki = 2 nM T82146 CWZY65 135754 Ki = 40 nM T82146 CRJ7K2 164456 Ki = 160 nM T82146 CI8NO1 3025917 EC50 = 340 nM T82146 C7AJR4 4433908 EC50 < 10000 nM T82146 CUL8F1 5354022 EC50 = 700 nM T82146 C8ES5G 6366138 EC50 = 200 nM T82146 C5EOB6 6366685 EC50 > 15 nM T82146 CGL71X 6366726 EC50 = 37 nM T82146 C5EON6 6366727 EC50 > 0.001 nM T82146 C62YGF 6366732 EC50 > 0.001 nM T82146 CK4UA6 6366733 EC50 > 0.001 nM T82146 CLF4M5 6366734 EC50 = 374 nM T82146 CA5GS8 6438168 EC50 > 0.001 nM T82146 C7C9SR 6439768 EC50 > 10000 nM T82146 CV6S9Y 6439770 EC50 = 0.4 nM T82146 C8WU1N 6440217 EC50 = 30 nM T82146 CG1S2D 6440346 EC50 = 0.4 nM T82146 C5LH2R 6441236 EC50 = 10 nM T82146 CJHW10 6441985 EC50 = 152 nM T82146 CHA3C2 6447986 EC50 = 12 nM T82146 C3F4GD 6447987 EC50 = 39 nM T82146 CEV62Y 6450532 EC50 = 47 nM T82146 C31YCL 9797765 Ki = 426 nM T82146 CBE62R 9799320 EC50 > 1000 nM T82146 CRK31P 9799442 EC50 = 1446 nM T82146 COP9S7 9799477 EC50 = 200 nM T82146 CENQ29 9799532 IC50 = 5 nM T82146 CSNI93 9799841 EC50 > 10000 nM T82146 CJ3ZM0 9801665 Ki = 1860 nM T82146 CX2HY4 9801929 EC50 > 10000 nM T82146 C8P4UD 9803186 Ki > 10000 nM T82146 CW7D0R 9810431 EC50 = 1604 nM T82146 CUJ14W 9819890 EC50 > 10000 nM T82146 CEK1O4 9820039 EC50 = 34 nM T82146 CQI49S 9820393 EC50 > 10000 nM T82146 C7R9JM 9820462 Ki = 1036 nM T82146 C2X3PS 9822318 EC50 = 22 nM T82146 C4WK5D 9824444 Ki = 4028 nM T82146 CI1P9A 9844563 Ki = 386 nM T82146 CQFA96 9845057 Ki > 9513 nM T82146 CE7D1J 9845382 IC50 = 4 nM T82146 CQ1ZH6 9847065 Ki > 10000 nM T82146 CA74MZ 9864886 IC50 = 3 nM T82146 CZK15S 9865215 Ki > 4000 nM T82146 C2ZY0W 9865875 EC50 > 1000 nM T82146 CB3NF2 9866384 Ki > 10000 nM T82146 CJ08SK 9867780 Ki > 10000 nM T82146 CAE0R3 9868664 Ki > 10000 nM T82146 CRC51S 9869157 Ki > 10000 nM T82146 CA0TS6 9884959 EC50 = 391 nM T82146 CSK5B8 9885521 EC50 > 1000 nM T82146 C6ZR5D 9885730 Ki = 10000 nM T82146 C3CS9R 9886082 EC50 > 10000 nM T82146 C5AD1H 9886137 Ki > 10000 nM T82146 CG3JR4 9887949 EC50 > 10000 nM T82146 C8V1ON 9888385 IC50 = 2 nM T82146 C90UXQ 9889347 Ki > 10000 nM T82146 C2WFX1 9905729 EC50 = 266 nM T82146 C2D9WJ 9906413 EC50 > 10000 nM T82146 C9AJZ7 9906514 EC50 = 24 nM T82146 C7E0IO 9907433 EC50 > 10000 nM T82146 CK9Z7I 9907650 IC50 = 310 nM T82146 COS0D4 9908099 Ki = 10000 nM T82146 CSF7G1 9908857 Ki = 10000 nM T82146 C0A3UZ 9911319 Ki > 10000 nM T82146 CSW2Y8 9929026 Ki > 1000 nM T82146 C9VEF0 9949645 EC50 = 2043 nM T82146 C6CI3S 9950957 EC50 > 10000 nM T82146 C0GLF2 9952045 Ki = 8566 nM T82146 CU46RB 9953712 Ki = 174 nM T82146 C6JLI1 9973307 EC50 > 10000 nM T82146 CV1A3K 9974457 EC50 > 1000 nM T82146 C63OUJ 9976842 EC50 > 1000 nM T82146 C05EXS 9998870 EC50 > 10000 nM T82146 CL7X4Y 9999621 EC50 > 10000 nM T82146 CM1BQ5 10003577 Ki = 8764 nM T82146 CZP71W 10022432 EC50 = 23 nM T82146 CN6LP5 10022568 EC50 > 10000 nM T82146 C6L0XH 10044201 Ki = 19 nM T82146 CN0Y1P 10044591 EC50 = 350 nM T82146 CE60FI 10065757 EC50 = 399 nM T82146 C2C0GJ 10066739 EC50 = 15 nM T82146 C4VU6T 10087372 EC50 > 10000 nM T82146 C8MG7C 10094345 IC50 > 3000 nM T82146 CZI69W 10112018 Ki > 10000 nM T82146 CPX6Q5 10115123 Ki > 10000 nM T82146 CSG68Q 10127015 IC50 = 2 nM T82146 C2S1QO 10158313 Ki > 10000 nM T82146 C72HLB 10172878 IC50 = 3.6 nM T82146 C15HAE 10194688 IC50 = 2 nM T82146 C9XS2G 10203771 Ki = 153 nM T82146 C0DS6Q 10223041 Ki > 10000 nM T82146 C7L4CJ 10225689 Ki > 10000 nM T82146 CKR51I 10225690 Ki > 10000 nM T82146 CVL1Q6 10227224 Ki = 151 nM T82146 CUV8S0 10249942 Ki = 10000 nM T82146 C3IHN5 10251128 IC50 = 331 nM T82146 CZY92F 10271982 Ki > 10000 nM T82146 COD29A 10272879 Ki > 10000 nM T82146 C2P8CN 10274512 Ki > 10000 nM T82146 C1LN6I 10274852 Ki > 10000 nM T82146 CCD7A5 10276434 Ki > 10000 nM T82146 CS6N3M 10298831 Ki > 10000 nM T82146 CY1J5M 10308975 EC50 = 144 nM T82146 C9D7QC 10314719 EC50 = 0.6 nM T82146 C7G6XH 10315687 EC50 = 3 nM T82146 CVQ7Z6 10316839 EC50 > 10000 nM T82146 C5LV9X 10358286 EC50 = 8 nM T82146 CUEF37 10362997 EC50 = 270 nM T82146 CG01ED 10383375 EC50 = 397 nM T82146 CW39AL 10384413 IC50 = 31 nM T82146 CJCA73 10385620 Ki = 53 nM T82146 C25HLM 10389354 Ki = 34 nM T82146 CXQ9S4 10450790 EC50 = 1016 nM T82146 CXA0N9 10458226 Ki = 490 nM T82146 CV7C4F 10478196 IC50 = 0.5 nM T82146 C0KZT7 10519016 Ki = 85 nM T82146 CY62NU 10523459 Ki = 20 nM T82146 CQR8K0 10524574 IC50 = 2 nM T82146 C5BXE0 10543210 EC50 > 1000 nM T82146 CUO1I2 10543981 Ki = 13 nM T82146 C6CWZ1 10545954 EC50 = 84 nM T82146 C26NJB 10547547 IC50 = 27 nM T82146 C9EBZ0 10572606 IC50 = 17 nM T82146 CKBI92 10619546 IC50 = 4.6 nM T82146 CS96IV 10619935 EC50 = 121 nM T82146 C2HXP8 10641611 Ki = 27 nM T82146 C1K6PS 10643199 IC50 = 150 nM T82146 CMH87P 10643692 EC50 > 10000 nM T82146 CZ2C5K 10663499 Ki = 200 nM T82146 C92TJP 10666483 Ki = 29 nM T82146 C9K4YM 10709275 EC50 > 1000 nM T82146 C1SNV6 10760998 Ki = 121 nM T82146 C9UFH8 10763649 Ki = 95 nM T82146 C2TJY4 10788561 Ki > 10000 nM T82146 CTI5N7 10789247 Ki = 72 nM T82146 CMXI39 10804037 EC50 = 230 nM T82146 CJ57NB 10916642 Ki = 2503 nM T82146 C8UG3F 10926235 EC50 > 500 nM T82146 CURV10 10926384 Ki > 10000 nM T82146 CWM7E2 10936808 Ki = 10000 nM T82146 CTB3E6 10937639 Ki = 10000 nM T82146 CF7DZ3 10938844 Ki = 10000 nM T82146 CG48CT 11025742 Ki = 10000 nM T82146 C6F1MJ 11079184 Ki = 10000 nM T82146 CO50RB 11080831 Ki = 10000 nM T82146 CV38KY 11167904 EC50 = 8 nM T82146 CT4HL6 11340230 IC50 > 1000000 nM T82146 CY6PJ9 11504066 EC50 = 10 nM T82146 CJH04T 11510627 EC50 = 20 nM T82146 CM34CL 11518525 EC50 = 1.9 nM T82146 C9NH8Y 11547131 EC50 = 3.6 nM T82146 CQAF21 11554936 EC50 = 4.7 nM T82146 CLID54 11569584 EC50 = 53 nM T82146 CQ8S3K 11627002 EC50 = 2.1 nM T82146 C41AJB 11634244 EC50 = 918 nM T82146 C3RMA0 11718697 EC50 = 353 nM T82146 C34NCO 11724776 EC50 > 1000 nM T82146 C0S9KJ 11740691 EC50 = 152 nM T82146 CFC0X5 11751490 IC50 = 19000 nM T82146 C0WA5F 11793407 EC50 = 17 nM T82146 CD5K4U 11799011 Ki > 10000 nM T82146 C7UWV3 12112296 EC50 = 91 nM T82146 CIQJ20 12112298 EC50 = 77 nM T82146 CQ9YE5 12358678 EC50 = 6 nM T82146 C7JSH9 13833722 EC50 = 330 nM T82146 C1M8SC 13833726 EC50 = 400 nM T82146 C7Z0YT 13833727 EC50 = 460 nM T82146 CT41DZ 14557465 EC50 = 2700 nM T82146 CN7CX1 14726558 IC50 = 21 nM T82146 C8DP6M 14776682 EC50 = 30 nM T82146 CQI17S 15160092 EC50 = 35 nM T82146 CNS9T8 15434197 Ki > 1000 nM T82146 CU8LV5 15951923 EC50 = 630.96 nM T82146 CDA7J9 15951925 EC50 < 10000 nM T82146 C5J3ZE 16661643 EC50 = 0.92 nM T82146 CX6L0G 16661644 EC50 = 0.22 nM T82146 C5GTA2 18507967 EC50 = 1100 nM T82146 CQYD01 18768139 EC50 = 2 nM T82146 CX3Q7D 20243100 EC50 = 1.4 nM T82146 C5MHX3 21217837 Ki = 148 nM T82146 CV1C4A 22226112 EC50 > 1000 nM T82146 CLV67T 22971725 EC50 = 6 nM T82146 CTE1N2 24748569 EC50 > 10000 nM T82146 CSTR97 25259041 EC50 = 158.49 nM T82146 C2G6QF 25259266 EC50 = 141.3 nM T82146 CO7M0D 44285104 EC50 = 550 nM T82146 CS7U6L 44285287 EC50 = 210 nM T82146 CBXN25 44307497 Ki = 280 nM T82146 CY0XR1 44307571 Ki = 710 nM T82146 CFTB98 44313143 Ki = 531 nM T82146 C4E1OW 44313513 Ki > 3000 nM T82146 C8W6JP 44314319 Ki = 32 nM T82146 C17LMT 44314320 Ki > 4000 nM T82146 C7U3IB 44316094 EC50 = 200 nM T82146 CRY69X 44316095 EC50 = 54 nM T82146 COX51B 44316155 EC50 = 260 nM T82146 C92VTZ 44316277 EC50 = 130 nM T82146 C8RM3G 44316292 EC50 = 4 nM T82146 C90NSH 44316354 EC50 = 20 nM T82146 CIVH74 44316525 Ki > 1000 nM T82146 CAP68W 44316543 Ki > 1000 nM T82146 CAI2Z5 44316544 Ki > 1000 nM T82146 C0YQ8H 44316756 Ki > 1000 nM T82146 C6Q1CA 44316796 Ki > 1000 nM T82146 CLK5H0 44316811 EC50 = 355 nM T82146 CFEG98 44321592 EC50 = 70 nM T82146 CK48CT 44321880 EC50 = 100 nM T82146 CID72B 44321881 EC50 = 1300 nM T82146 CXV0B4 44321951 EC50 = 1500 nM T82146 C1KUN0 44325759 Ki > 1000 nM T82146 CLB6X7 44325767 Ki > 1000 nM T82146 C39LIO 44325862 Ki > 10000 nM T82146 CK6JC0 44338117 Ki > 10000 nM T82146 CP51SQ 44338305 Ki > 10000 nM T82146 CG6H2T 44353335 Ki > 10000 nM T82146 CW0T6K 44353336 Ki > 10000 nM T82146 C8K0AB 44353347 Ki > 10000 nM T82146 C3DYE9 44353422 Ki > 10000 nM T82146 C5DTY3 44353441 Ki > 10000 nM T82146 C2M8TN 44353456 Ki > 10000 nM T82146 CVKA40 44353466 Ki > 10000 nM T82146 C8J5SA 44353480 Ki > 1000 nM T82146 CIB15X 44353481 Ki > 10000 nM T82146 C3MY4C 44364348 Ki = 860 nM T82146 CY9XP2 44366042 EC50 > 10000 nM T82146 CT3S5O 44377822 EC50 = 4 nM T82146 C5QRI4 44401302 IC50 = 1200 nM T82146 CJVG73 44459626 EC50 = 2000 nM T82146 CR5SI0 44476535 EC50 > 10000 nM T82146 CP4DM5 44581289 EC50 = 10 nM T82146 C8UHG5 45270032 IC50 = 40 nM T82146 CUD91T 49862248 EC50 > 10000 nM T82146 CFO23H 56837193 IC50 > 10000 nM T82146 CZE4U3 60162553 IC50 = 1300 nM T82146 C9G4IT 60729785 EC50 = 109.2 nM T82146 CZ38NM 69588033 EC50 = 6 nM T82146 CVY3G8 71247311 IC50 > 10000 nM T82146 CN03UB 71568951 EC50 = 383 nM T82146 CX9EA0 71568952 EC50 = 847.2 nM T82146 C4GRK9 71571262 EC50 = 98.9 nM T82146 C1WA6T 118142048 IC50 > 10000 nM T82146 C6IX2E 118142057 IC50 = 1400 nM T82146 C7D3AT 121429517 IC50 > 10000 nM T82146 CB9GP5 122235238 IC50 = 7200 nM T82146 C7CZG3 134131811 IC50 > 10000 nM T82146 CP1U5T 134132295 IC50 > 10000 nM T82146 CB6C7O 134133110 IC50 > 10000 nM T82146 C2Z0DR 134133677 IC50 > 10000 nM T82146 C0VX8Q 134135363 IC50 = 4100 nM T82146 C1UVG3 134137057 IC50 = 800 nM T82146 C60HIA 134137870 IC50 > 10000 nM T82146 CGO9C7 134138123 IC50 > 10000 nM T82146 CH9VS2 134138409 IC50 > 10000 nM T82146 CL85MU 134139004 IC50 = 5600 nM T82146 CK5CZ8 134139028 IC50 > 10000 nM T82146 CR7J9Q 134139617 IC50 > 10000 nM T82146 CJQ8O6 134139787 IC50 = 6200 nM T82146 CH4O7X 134140416 IC50 > 10000 nM T82146 C7TMP3 134140572 IC50 > 10000 nM T82146 CR0CX8 134141317 IC50 = 1100 nM T82146 C5Y0XG 134141341 IC50 > 10000 nM T82146 CS4V8O 134141363 IC50 > 10000 nM T82146 C61WKA 134142331 IC50 = 7600 nM T82146 CR69NQ 134142378 IC50 > 10000 nM T82146 C8FS0G 134142941 IC50 > 10000 nM T82146 CKD1S2 134144175 IC50 > 10000 nM T82146 C8QNS0 134145062 IC50 = 2700 nM T82146 C4AO0F 134145297 IC50 = 4400 nM T82146 CCWS64 134145922 IC50 > 10000 nM T82146 C68HUB 134146033 IC50 > 10000 nM T82146 C6XZY1 134147284 IC50 = 3500 nM T82146 CY4R8J 134147557 IC50 = 4500 nM T82146 C3AHY8 134147641 IC50 > 10000 nM T82146 C9LPU5 134148070 IC50 = 4200 nM T82146 CLC9U8 134148522 IC50 = 3800 nM T82146 CT6GX8 134148836 IC50 > 10000 nM T82146 CV1MC9 134149320 IC50 > 10000 nM T82146 C07QGW 134149538 IC50 = 7700 nM T82146 CJ75KB 134149807 IC50 > 10000 nM T82146 CPO31X 134150617 IC50 = 1900 nM T82146 COC3J0 134151576 IC50 = 1400 nM T82146 CO12JS 134152058 IC50 = 9100 nM T82146 C0MNC7 134152441 IC50 > 10000 nM T82146 C6B5DW 134154628 IC50 = 6800 nM T82146 CHIZ89 134155284 IC50 > 10000 nM T82146 C3PGZ2 134155420 IC50 = 6800 nM T82146 C8HJE4 134156268 IC50 = 8400 nM T82146 CTV56P 134156567 IC50 > 10000 nM T82146 CVER01 134157830 IC50 = 5700 nM T82146 C6L4GM 135949402 EC50 = 91 nM T82146 C5L6AU 136126668 EC50 > 1000 nM T82146 CN5MO3 136126669 EC50 > 1000 nM T82146 CJ5EH7 136126670 EC50 > 1000 nM T82146 CI4CG1 136126671 EC50 > 1000 nM T82146 C2FK0D 145964346 EC50 = 168 nM T82146 C1J4DV 145965542 EC50 = 11 nM T82146 CRKW68 145966900 EC50 > 10000 nM T82146 CM13TV 145967217 EC50 = 85 nM T82146 C4MY5N 145967331 EC50 = 4.4 nM T82146 CC05VW 145970742 EC50 = 67 nM T82146 CSY61C 145971359 EC50 = 120 nM T82146 CD35WU 145971426 EC50 = 47 nM T82146 C3ZI2W 145971858 EC50 = 7.4 nM T82146 C4GEX7 145973883 EC50 = 60 nM T82146 C4E0NZ 145975370 EC50 = 279 nM T82146 CDBR75 145976745 EC50 = 1.4 nM T82146 CIMO76 145977706 EC50 = 15 nM T82146 CYIG73 145977797 EC50 = 422 nM T82146 C2A1UC 10429766 EC50 = 209 nM T82146 D09RRF 11530459 EC50 = 501.19 nM T82146 D0F8CC 10090192 EC50 = 46 nM T82146 D0G6JM 5289501 EC50 = 2 nM T82146 D0P0PP 10044792 IC50 = 22000 nM T82146 D0Q0IR 177238 IC50 = 3 nM T82146 D0Q9FZ 6442223 EC50 = 192 nM T82146 D0RD0R 2126 EC50 = 13 nM T96435 C7FMI4 99148 IC50 = 6100 nM T96435 C9IDX7 1007757 IC50 = 17600 nM T96435 C61MKS 1026589 IC50 = 23500 nM T96435 CMC4W7 1027199 IC50 = 15800 nM T96435 C98GRU 1216550 IC50 = 3542 nM T96435 CBU57A 1330989 IC50 = 2385 nM T96435 C8ZOB9 1919138 IC50 = 28400 nM T96435 C81SRX 2243305 IC50 = 20800 nM T96435 C54EYV 4087515 IC50 = 15000 nM T96435 CT43SB 4553749 IC50 = 47900 nM T96435 CCQN16 6874616 IC50 = 18400 nM T96435 CFZ8J6 9616054 IC50 = 14000 nM T96435 CD78KT 10089837 IC50 = 21200 nM T96435 C63ITL 10387923 IC50 > 100000 nM T96435 CT0O5K 10634145 IC50 > 31600 nM T96435 C5DZ7R 23829354 IC50 = 1856 nM T96435 CNS64M 23848602 IC50 > 50000 nM T96435 CL7RK9 25191039 IC50 = 2710 nM T96435 CI0OD8 56598331 IC50 = 9200 nM T96435 CWZ8V1 57390914 IC50 = 21800 nM T96435 CZ7L3W 57394433 IC50 > 100000 nM T96435 C9HYB8 57394434 IC50 = 21200 nM T96435 C9C6SM 57396194 IC50 > 100000 nM T96435 CBT1R5 57398002 IC50 > 100000 nM T96435 C32LRX 57399658 IC50 > 100000 nM T96435 C3H4ZO 57399659 IC50 = 27200 nM T96435 CN49BK 57399660 IC50 > 100000 nM T96435 CO7CG3 57403163 IC50 = 15500 nM T96435 C8V5MQ 66552710 IC50 = 39500 nM T96435 CTA4V2 66552711 IC50 = 29600 nM T96435 C1GKU3 70691637 IC50 = 9730 nM T96435 C3C7LX 71451488 IC50 = 1080 nM T96435 C5WYX6 71456815 IC50 > 50000 nM T96435 CX5U1W 71460502 IC50 = 1175 nM T96435 CFS3K0 71460503 IC50 = 1735 nM T96435 CXVJ86 71462210 IC50 > 50000 nM T96435 C6OY4U 71462211 IC50 > 50000 nM T96435 C3UO4R 127046748 IC50 = 3300 nM T96435 C3H4RT 134131655 IC50 = 16400 nM T96435 CMYX73 134132415 IC50 = 8000 nM T96435 CNAG53 134134717 IC50 = 9100 nM T96435 CUZ9N1 134136743 IC50 = 15300 nM T96435 C59OJM 134141604 IC50 = 6200 nM T96435 CV3PO2 134144907 IC50 = 8500 nM T96435 C0OXC4 134146531 IC50 = 4900 nM T96435 CAY2G3 134151404 IC50 = 12400 nM T96435 CJM61X 134153461 IC50 = 6400 nM T96435 C0G2CU 134155303 IC50 = 26600 nM T96435 C6GE0K 134155989 IC50 = 7100 nM T96435 C63PGS 134156985 IC50 = 7600 nM T96435 CY0RC7 134157144 IC50 = 3500 nM T96435 CKC1Z2 135609425 IC50 = 20700 nM T96435 CL4S2M 155566367 IC50 = 1520 nM T96435 D0Y7OI 11563133 Ki = 930 nM T30790 D00AXJ 4189 IC50 = 100000 nM T30790 D0EV8E 3198 IC50 = 17000 nM T30790 D0W8XT 60663 IC50 = 52100 nM T30790 CKA06J 2740687 IC50 = 57000 nM T30790 CADH79 2881318 IC50 = 75000 nM T30790 C2LP4Z 2884116 IC50 = 47000 nM T30790 C2HCI5 9586645 IC50 = 69900 nM T30790 C1O9VD 45874974 IC50 = 48000 nM T30790 CGQ5N4 71603470 IC50 < 100 nM T30790 C7YAQ1 75202944 IC50 = 104 nM T30790 CZFT61 90184724 IC50 = 440 nM T30790 C6XZ9N 132547220 IC50 = 26 nM T30790 CC1I2J 132547221 IC50 = 42000 nM T30790 CD6K5Z 134153740 IC50 = 100000 nM T30790 C9X4CB 145960410 IC50 = 89000 nM T30790 CW3KH6 145960508 IC50 = 47000 nM T30790 C21KDB 145960529 IC50 = 75000 nM T30790 C46WAU 145960617 IC50 = 33000 nM T30790 C2JIU0 145960707 IC50 = 29000 nM T30790 C58RAK 145961304 IC50 = 54000 nM T30790 CK76EL 145961532 IC50 = 79000 nM T30790 C1FI5B 145961536 IC50 = 49000 nM T30790 CBCT61 145961548 IC50 = 45000 nM T30790 C0A6LE 145961674 IC50 = 42000 nM T30790 CSL52Y 145961931 IC50 = 42000 nM T30790 C9PMX3 145962134 IC50 = 30000 nM T30790 CD3B1Y 145962241 IC50 = 40000 nM T30790 CC71JG 145962327 IC50 = 48000 nM T30790 CEN9W7 145962441 IC50 = 32000 nM T30790 CS1N9B 145962471 IC50 = 55000 nM T30790 CTZF07 145962595 IC50 = 60000 nM T30790 C5U9PO 145962607 IC50 = 33000 nM T30790 C4BQ3Y 145962619 IC50 = 36000 nM T30790 CA46MP 145963236 IC50 = 105000 nM T30790 C2V6AM 145963278 IC50 = 89000 nM T30790 CX76NP 145963560 IC50 = 55000 nM T30790 C6NF2H 145963592 IC50 = 58000 nM T30790 CE16PU 145963603 IC50 = 42000 nM T30790 D0JV2P 2455 IC50 = 2800 nM T82297 D01KKQ 135400182 IC50 = 22 nM T82297 D0SV8E 126941 IC50 = 211 nM T82297 D0Y4GO 135410875 IC50 = 60 nM T82297 CPM3L5 67092576 IC50 = 17.5 nM T82297 CTK64O 67092918 IC50 = 54.3 nM T82297 C9Z4ES 135567027 IC50 = 5.6 nM T82297 CF39AI 135567029 IC50 = 0.17 nM T82297 C8N7ES 135567030 IC50 = 0.43 nM T82297 CFE2O7 135567034 IC50 = 0.34 nM T82297 C8KVP5 135567035 IC50 = 654 nM T82297 CSQX75 135567163 IC50 = 0.62 nM T82297 CQF8P5 135800109 IC50 = 5.6 nM T82297 CR7UY3 136044173 IC50 = 3.6 nM T82297 C0Q5FI 136044174 IC50 > 1000 nM T82297 CGX68Y 136044175 IC50 > 1000 nM T82297 C4C9FN 136044176 IC50 = 347 nM T82297 CIPD35 136044177 IC50 > 1000 nM T82297 CZG8W6 136059167 IC50 = 0.51 nM T82297 CZC95Y 136059168 IC50 = 37.41 nM T82297 CG2ID9 136059169 IC50 > 1000 nM T82297 C2WH0S 136059178 IC50 > 1000 nM T82297 CB3GL7 136059191 IC50 = 839.1 nM T82297 CCHG08 136059192 IC50 = 18.8 nM T82297 CUF8R1 155515541 IC50 = 0.93 nM T82297 CMKA64 155517044 IC50 = 1.57 nM T82297 CCL3Y9 155518053 IC50 = 0.19 nM T82297 C91SVN 155519837 IC50 = 2.59 nM T82297 CT70WU 155530762 IC50 = 0.75 nM T82297 CX42MF 155532591 IC50 = 0.34 nM T82297 CFU98A 155534971 IC50 = 0.53 nM T82297 C6S7OC 155548982 IC50 = 3.87 nM T82297 CX3K8F 155549935 IC50 = 1.6 nM T82297 CJ0MK5 155554671 IC50 = 0.44 nM T82297 CYQ0I9 155555353 IC50 = 0.45 nM T91598 D0E3TC 44259 IC50 = 0.584 nM T91598 C3VRO9 44557921 IC50 > 10000 nM T91598 CV63UL 67240318 IC50 > 10000 nM T01249 D0I6LH 107985 IC50 = 30900 nM T01249 C1EXW3 334509 IC50 = 900 nM T01249 C6S1MX 661498 IC50 = 19 nM T01249 CFJG92 662681 IC50 = 1880 nM T01249 CWM2C9 662768 IC50 = 704 nM T01249 CMP64A 662931 IC50 = 79 nM T01249 CKF21I 663002 IC50 = 440 nM T01249 CC7FI1 663393 IC50 = 419 nM T01249 C7RG1V 860112 IC50 = 920 nM T01249 CBT19P 931337 IC50 > 10000 nM T01249 C5MLV1 932337 IC50 = 619 nM T01249 CT1G9Q 933867 IC50 = 271 nM T01249 C3MTV8 934087 IC50 = 1030 nM T01249 CL3AD2 934157 IC50 = 282 nM T01249 CSN45R 935908 IC50 = 2610 nM T01249 CI40SY 936290 IC50 = 449 nM T01249 C2RCQ7 936793 IC50 = 469 nM T01249 C72PNM 936863 IC50 = 449 nM T01249 CS07QM 937168 IC50 = 592 nM T01249 CSL5H2 937750 IC50 = 505 nM T01249 CE0HL9 938350 IC50 = 204 nM T01249 CJI6F4 938542 IC50 = 291 nM T01249 COZ5R0 977367 IC50 = 144 nM T01249 C96QVH 1070528 IC50 = 370 nM T01249 C6X1AS 1091495 IC50 = 3200 nM T01249 C27OFH 1091496 IC50 = 2500 nM T01249 CILC18 1265686 IC50 = 620 nM T01249 CK07JQ 1479155 IC50 = 57 nM T01249 CUH62Z 1591626 IC50 = 520 nM T01249 C3RM0Z 1855778 IC50 = 600 nM T01249 C62EKX 1863824 IC50 = 190 nM T01249 C0YNB6 1992853 IC50 = 164 nM T01249 CS5R4F 2857183 IC50 = 1910 nM T01249 CQ7M8T 2857275 IC50 = 940 nM T01249 C4SRX1 2894916 IC50 = 1100 nM T01249 C5O2GC 2951229 IC50 = 1500 nM T01249 CCF70I 2958654 IC50 = 1200 nM T01249 C10PMY 2960286 IC50 = 810 nM T01249 CVEG10 2960577 IC50 = 910 nM T01249 C0HCQ6 2960766 IC50 = 990 nM T01249 C5CIN6 2988522 IC50 = 208 nM T01249 CNSC26 2988623 IC50 = 1200 nM T01249 C6XZ8B 2988707 IC50 = 410 nM T01249 C32UCQ 3163969 IC50 = 20 nM T01249 C2BYN7 3700079 IC50 = 2100 nM T01249 CZ6UC7 4250909 IC50 > 100000 nM T01249 C8R4LT 4886428 IC50 = 200 nM T01249 C6GV0E 4902357 IC50 = 170 nM T01249 CJTZ67 4972973 IC50 = 1500 nM T01249 C64IVU 5306520 IC50 = 691 nM T01249 C06KNI 5311821 IC50 = 1031 nM T01249 C8ANX1 6456513 IC50 = 1100 nM T01249 CG9EN3 6462251 IC50 = 450 nM T01249 C8OF1Y 6471263 IC50 = 6973 nM T01249 CFOM17 6473084 IC50 = 7456 nM T01249 CA3VG6 6500352 IC50 = 840 nM T01249 C4EDF0 8033802 IC50 = 177 nM T01249 CR90ZW 8033823 IC50 > 10000 nM T01249 CJS15D 9152594 IC50 > 100000 nM T01249 CKD6B7 9566630 IC50 = 370 nM T01249 CFQ46Z 11223729 IC50 = 1400 nM T01249 CZON96 16035660 IC50 = 2800 nM T01249 C92GOW 16414816 IC50 = 190 nM T01249 C9REB8 16416765 IC50 = 314 nM T01249 C6S8VA 16421196 IC50 = 401 nM T01249 CWO05C 16423079 IC50 = 1700 nM T01249 CM0Q3L 16457425 IC50 = 1100 nM T01249 C67OHE 16457434 IC50 = 730 nM T01249 C0QXV3 16460104 IC50 = 8600 nM T01249 CA6ED8 16460189 IC50 = 3400 nM T01249 C3S5RV 16763116 IC50 = 346 nM T01249 CSUI08 16764758 IC50 = 357 nM T01249 CD0A6I 16764760 IC50 = 332 nM T01249 C95ORB 16995008 IC50 > 100000 nM T01249 CU1D8C 16995210 IC50 > 100000 nM T01249 C9XA1Q 17014838 IC50 = 1300 nM T01249 CVU4Q8 17014844 IC50 = 360 nM T01249 CTBZ96 17014847 IC50 = 780 nM T01249 CW5UL9 17014889 IC50 = 2100 nM T01249 C46KQZ 17015681 IC50 = 860 nM T01249 C8PIE9 17079438 IC50 = 850 nM T01249 C10ZXL 17248373 IC50 = 1400 nM T01249 C94SEW 17587429 IC50 = 550 nM T01249 CFN0O1 17590104 IC50 = 277 nM T01249 CKYZ04 17591943 IC50 = 233 nM T01249 CGN87A 17593912 IC50 = 670 nM T01249 CYF81V 17593955 IC50 = 328 nM T01249 C6LOX7 17720024 IC50 = 990 nM T01249 CC38SV 18891468 IC50 = 580 nM T01249 COJ1M9 18891516 IC50 = 1400 nM T01249 CNHT84 18891564 IC50 = 2200 nM T01249 CE1N8U 21319368 IC50 = 1200 nM T01249 CMZ8W7 24824904 IC50 = 2064 nM T01249 CXJP28 24824926 IC50 = 1021 nM T01249 C47LCS 24824940 IC50 = 505 nM T01249 CKI60C 25020906 IC50 = 227 nM T01249 CQTP54 25020907 IC50 = 602 nM T01249 CJB6U1 25020909 IC50 = 276 nM T01249 CJ2MR1 25020910 IC50 = 95 nM T01249 C3NP5G 25239884 IC50 = 1168 nM T01249 CS9EW2 27772148 IC50 = 660 nM T01249 CK92VU 41448380 IC50 = 1215 nM T01249 CCJ8I9 41448381 IC50 = 204 nM T01249 CJ3FV7 41905062 IC50 = 5610 nM T01249 CBW10U 56692515 IC50 > 10000 nM T01249 CEC4K9 66849498 IC50 > 10000 nM T01249 COW29T 71521050 IC50 = 240 nM T01249 C5ZX3L 121269983 IC50 = 165 nM T01249 C15AZT 121269984 IC50 = 73 nM T01249 CQ1M2X 121269987 IC50 = 240 nM T01249 COL92V 121269988 IC50 = 41 nM T01249 CT2PF7 121269992 IC50 = 250 nM T01249 COP3W5 121269993 IC50 = 49 nM T01249 CI46EN 121269994 IC50 = 96 nM T01249 C34UBK 121269996 IC50 = 190 nM T01249 CI56SW 121269999 IC50 = 185 nM T01249 C8XP0L 121270000 IC50 = 19 nM T01249 CO2C6V 121270009 IC50 = 95 nM T01249 C3CJ9E 121270013 IC50 = 75 nM T01249 CZUW50 121270021 IC50 = 331 nM T01249 CJEK18 121270024 IC50 = 21 nM T01249 CT8YZ3 121270027 IC50 = 34 nM T01249 C5LBJ3 121270029 IC50 = 1450 nM T01249 C4HRI5 121270030 IC50 = 74 nM T01249 CDH4O3 121270031 IC50 = 133 nM T01249 C3PM0I 121270037 IC50 = 85 nM T01249 C7TUW8 127025699 IC50 = 27 nM T01249 C29BQZ 127025700 IC50 = 206 nM T01249 C27WMP 127025701 IC50 = 248 nM T01249 CK9OR6 127026287 IC50 = 82 nM T01249 COK8Q9 127026288 IC50 = 46 nM T01249 CU32KG 127026289 IC50 = 47 nM T01249 C5VB0P 127026290 IC50 = 205 nM T01249 CET7F2 127026557 IC50 = 12000 nM T01249 CJI5X8 127026587 IC50 = 529 nM T01249 CKZ47F 127026889 IC50 = 22000 nM T01249 C9WJ7T 127026890 IC50 = 46 nM T01249 C8V2BX 135445400 IC50 = 1500 nM T01249 CP8C7U 135491346 IC50 = 2200 nM T01249 CRNJ96 135491350 IC50 = 1400 nM T01249 C0QB2H 135491367 IC50 = 1100 nM T01249 C1CP9N 135504353 IC50 = 1000 nM T01249 C84HVO 135541817 IC50 = 240 nM T01249 CEWX17 135602362 IC50 = 1500 nM T01249 CT1DZ8 135644892 IC50 = 1500 nM T01249 C0XWZ3 135644949 IC50 = 1100 nM T01249 C86HMY 137631644 IC50 > 10000 nM T01249 CI2ZY5 137633527 IC50 = 170 nM T01249 C2W0XU 137634059 IC50 = 350 nM T01249 C6N0GZ 137634805 IC50 = 1700 nM T01249 C31ZMA 137634968 IC50 = 34 nM T01249 C3CH8A 137635889 IC50 = 980 nM T01249 CZGD21 137635977 IC50 = 453 nM T01249 CO03MP 137636956 IC50 = 558 nM T01249 C9T1GM 137637534 IC50 = 65 nM T01249 C3NY1P 137637959 IC50 > 100000 nM T01249 CG1R3J 137638393 IC50 = 850 nM T01249 CTQG12 137638565 IC50 = 19 nM T01249 CTR6Q5 137639207 IC50 = 8400 nM T01249 C87SAX 137639947 IC50 = 1100 nM T01249 CS01XB 137639970 IC50 = 220 nM T01249 CG42MS 137640592 IC50 = 1000 nM T01249 C5MC4A 137640618 IC50 = 3200 nM T01249 CT0H6L 137643410 IC50 > 100000 nM T01249 C8GAZ9 137643773 IC50 = 502 nM T01249 C27XST 137644275 IC50 = 1366 nM T01249 CJU8F5 137644327 IC50 = 250 nM T01249 C4KJC8 137646447 IC50 > 100000 nM T01249 CT8W2A 137647511 IC50 = 530 nM T01249 C23SIL 137647575 IC50 > 10000 nM T01249 CA87ZL 137647837 IC50 = 280 nM T01249 C4T0RF 137648602 IC50 = 25 nM T01249 C21DXS 137649574 IC50 > 10000 nM T01249 CX6DL4 137649715 IC50 = 36 nM T01249 CO6Y7Z 137649899 IC50 = 260 nM T01249 CST72C 137651039 IC50 = 890 nM T01249 CMN4G5 137653001 IC50 = 258 nM T01249 CPIB08 137653673 IC50 = 41 nM T01249 C4UZJ3 137654315 IC50 = 6505 nM T01249 CJ3X0E 137656590 IC50 > 10000 nM T01249 CL79NI 137657375 IC50 = 1600 nM T01249 C10BOF 137659469 IC50 = 51 nM T01249 CAES91 137659877 IC50 = 38 nM T01249 CK37AQ 137660176 IC50 = 1500 nM T01249 C0UZF4 137661209 IC50 > 10000 nM T01249 CE2QU7 137661311 IC50 = 1600 nM T01249 CF3RQ7 137662061 IC50 = 1800 nM T01249 CILU71 137662287 IC50 = 2600 nM T98390 D08EYQ 448281 IC50 = 0.44 nM T98390 CE1H5V 1382255 IC50 = 62000 nM T98390 C8P2UD 24827309 Ki = 7.5 nM T98390 CRS26D 24827437 Ki = 6.5 nM T98390 CD0ME8 24827440 Ki = 7 nM T98390 CG6WS4 24827547 Ki = 5.2 nM T98390 C0SEG1 24827658 Ki = 5.2 nM T98390 CUYB68 24827661 Ki = 6.6 nM T98390 CYP60C 24827781 Ki = 0.7 nM T98390 C79VFM 24827784 Ki = 920 nM T98390 C01XOT 24827913 Ki = 800 nM T98390 C9A0HU 24828308 Ki = 300 nM T98390 C5ESN2 24828309 Ki = 300 nM T98390 C7NS5H 24828310 Ki = 3000 nM T98390 CH8IC5 24828443 Ki > 10000 nM T98390 C02ZBM 24828444 Ki > 10000 nM T98390 CI0A7J 24828445 Ki = 8000 nM T98390 C7W5MA 24828578 Ki > 10000 nM T98390 C6FGD3 24828579 Ki > 10000 nM T98390 C98THQ 24828580 Ki > 10000 nM T98390 C74JBV 24829232 Ki > 10000 nM T98390 CP2LY7 25033280 Ki = 1.5 nM T98390 C4YKQ1 25033281 Ki = 7.1 nM T98390 CG75AN 44377126 Ki = 86 nM T98390 C06HJB 44446952 Ki = 1.5 nM T98390 CNK7X5 44446953 Ki = 90 nM T98390 CEB78N 44446954 Ki = 14 nM T98390 CMO78A 44446956 Ki = 1.5 nM T98390 CV6H2M 44446957 Ki = 1.3 nM T98390 CF4KE1 44446959 Ki = 2.2 nM T98390 CW9C0E 44446960 Ki = 2.4 nM T98390 CQB5M0 44446963 Ki = 37 nM T98390 C94POY 44446965 Ki = 2.2 nM T98390 CBX2U9 44446967 Ki = 0.9 nM T98390 CRZ6B3 44446968 Ki = 5.8 nM T98390 CY9O4I 44446969 Ki = 2.2 nM T98390 C4PQ7D 44446970 Ki = 6 nM T98390 C96KIY 44446972 Ki = 2.4 nM T98390 CK1EM5 44446974 Ki = 2.7 nM T98390 C4V6RZ 44446975 Ki = 2.5 nM T98390 CBL9E6 44446976 Ki = 2 nM T98390 CVYX54 44446979 Ki = 0.85 nM T98390 CAI9Z6 44446980 Ki = 35 nM T98390 C86KVP 44446984 Ki = 84 nM T98390 CXP2V4 44450296 Ki = 220 nM T98390 C29JUG 44450311 Ki = 0.4 nM T98390 C29YXI 44450312 Ki = 1.25 nM T98390 CC2IS3 44454957 Ki = 65 nM T98390 C1ESI2 44454959 Ki = 2.4 nM T98390 C8L0MV 44454960 Ki = 1.8 nM T98390 CBG6T0 44454987 Ki = 1.6 nM T98390 CN7UW3 44455013 Ki = 1.8 nM T98390 CC5L7S 44455015 Ki = 2300 nM T98390 C6KDT1 44455016 Ki = 1.4 nM T98390 CF4ML7 44455018 Ki = 6.9 nM T98390 CZI6S1 44455047 Ki = 320 nM T98390 C3UF6E 44455406 Ki = 860 nM T98390 CJG71N 44455407 Ki = 550 nM T98390 C0IR5W 44455428 Ki = 420 nM T98390 C62KSV 44455429 Ki = 84 nM T98390 CR9WL2 44455430 Ki = 1.4 nM T98390 CGH0S7 54589400 IC50 > 100000 nM T98390 D05JBC 98888 IC50 = 57000 nM T98390 D0N4RO 44377139 Ki = 1400 nM T98390 D0P0MP 24827312 Ki = 0.13 nM T31935 D02UDJ 71077 Ki = 22000000 nM T31935 D02WFK 6234 Ki = 4400000 nM T31935 D03KEK 3765 Ki = 5800000 nM T31935 D09PUL 5950 Ki = 2800000 nM T31935 D0DZ3X 145742 Ki = 1600000 nM T31935 D0EP8X 10413 Ki = 65000000 nM T31935 D0FD0H 564 Ki = 35000000 nM T31935 D0M8AB 750 Ki = 5100000 nM T31935 D0XB8P 247 Ki = 1900000 nM T31935 D01WZG 586 Ki = 3200000 nM T31935 D09DLP 1646 Ki = 7100000 nM T31935 D0C9XA 119 Ki = 4000000 nM T31935 D0L4VI 5862 Ki = 46000000 nM T31935 D0M0UT 72390 Ki = 46000000 nM T31935 CRO5W2 588 Ki = 15000000 nM T31935 C2Z6BN 1018 Ki = 18000000 nM T31935 CLE87P 7419 Ki = 12000000 nM T31935 C9GIQ1 10444 Ki = 44000000 nM T31935 CF7HS5 31268 Ki = 38000000 nM T31935 CCB1F7 65098 Ki = 46000000 nM T31935 C5X2WA 71563 Ki = 100000000 nM T31935 CB6C2V 80283 Ki = 35000000 nM T31935 CTJ0Y3 93176 Ki = 7900000 nM T31935 CZ8UM4 157018 Ki = 4800000 nM T31935 CYK45X 439227 Ki = 11000000 nM T31935 C7JI5G 439575 Ki = 100000000 nM T31935 CA37FE 440014 Ki = 3300000 nM T31935 CNY8E4 440015 Ki = 30000000 nM T31935 C4V5ME 440575 Ki = 37000000 nM T31935 CF43JH 449215 Ki = 7400000 nM T31935 C04HXS 640091 Ki = 50000000 nM T31935 C34NKT 736316 Ki = 2500000 nM T31935 CK0UF5 5288725 Ki = 2200000 nM T31935 CX19WB 11073435 Ki = 2700000 nM T31935 D00BFT 16486 Ki = 1800000 nM T31935 D01BCI 71080 Ki = 19000000 nM T31935 D02YMI 5810 Ki = 9000000 nM T31935 D03ZKN 67701 Ki = 1300000 nM T31935 D06DRS 8082 Ki = 54000000 nM T31935 D08JUG 6119 Ki = 23000000 nM T31935 D0AC2H 3773 Ki = 2300000 nM T31935 D0AH1H 763 Ki = 1500000 nM T31935 D0C6IE 1123 Ki = 7800000 nM T31935 D0I8SK 6306 Ki = 37000000 nM T31935 D0O1QK 75725 Ki = 2200000 nM T31935 D0T6GM 5951 Ki = 35000000 nM T31935 D0TE9B 8988 Ki = 1200000 nM T31935 D0W4MZ 6106 Ki = 100000000 nM T31935 D0W8SX 239 Ki = 2400000 nM T31935 D0YF9S 1088 Ki = 1900000 nM T78656 D0Z6UC 5358 Ki = 25.7 nM T78656 D09GHO 5311258 Ki = 1.6 nM T78656 D02ZSO 6426760 IC50 = 3800 nM T78656 D0Q2JS 10436045 Ki = 3.162 nM T78656 D0YP7L 6604889 Ki < 3162.28 nM T78656 C0QCK1 6918455 Ki < 1000 nM T78656 CW0ZE5 6918542 Ki = 2500 nM T78656 CD0Z4I 6918648 Ki = 251.19 nM T78656 CUD06Z 9796627 Ki = 29 nM T78656 C4N3JX 9798021 Ki = 5.1 nM T78656 CWOS30 9817810 Ki = 47 nM T78656 CO13NK 9840850 Ki = 8.2 nM T78656 CNCK78 9862256 Ki = 3.9 nM T78656 CCJZ06 9863365 Ki = 3.1 nM T78656 CB1F0C 9867475 Ki = 570 nM T78656 CJW1P5 9888494 Ki < 10000 nM T78656 C3J8GU 9892409 Ki < 1000 nM T78656 C78MDV 9913554 Ki = 316.23 nM T78656 C4UYZ7 9927441 Ki = 770 nM T78656 CWO45F 9935387 Ki = 199.53 nM T78656 CYH3R7 9947817 Ki = 5.5 nM T78656 C63EWV 9950390 Ki = 3.9 nM T78656 CW83MT 10000386 Ki = 2.3 nM T78656 CK18LT 10020895 Ki = 7.6 nM T78656 CMWD23 10198756 Ki = 23 nM T78656 CQ7ND4 10220230 Ki = 100 nM T78656 C4NGF1 10220244 Ki = 100 nM T78656 C4Q2SH 10249573 Ki < 10000 nM T78656 CMRA02 10257042 Ki < 3162.28 nM T78656 CDH1O2 10308815 Ki = 9.5 nM T78656 C9IAV3 10346043 Ki > 10000 nM T78656 C4TPN1 10413595 Ki > 7943.28 nM T78656 CD7U5I 10433930 Ki > 10000 nM T78656 CBAY90 10445946 Ki = 5 nM T78656 CHE80N 10573876 Ki < 5011.87 nM T78656 CO23YX 10597140 Ki < 10000 nM T78656 C8MHZ9 10835110 Ki < 3162.28 nM T78656 CD4WJ3 10861816 Ki = 30 nM T78656 C8HN1F 10872581 Ki = 7.7 nM T78656 CN5A4L 10873909 Ki = 75 nM T78656 CN5JM4 10880608 Ki = 21 nM T78656 C8OYI0 10891048 Ki = 220 nM T78656 C1RAP3 10904295 Ki = 13 nM T78656 C0Q7GV 10915350 Ki = 11 nM T78656 CGJD40 10925076 Ki = 14 nM T78656 CZN8J0 10925382 EC50 = 11 nM T78656 C5X1OQ 10926112 Ki = 5.8 nM T78656 CRM8B3 10934159 Ki = 45 nM T78656 CQ0Z3K 10945589 Ki = 35 nM T78656 CWE3C9 10946905 Ki = 8.7 nM T78656 CVX54H 10959868 Ki = 18 nM T78656 C7GHU5 10970604 Ki = 11 nM T78656 C86GIP 10971452 Ki = 4.1 nM T78656 CZP7F0 10991087 Ki = 13 nM T78656 CPU5J4 10991464 Ki = 13.5 nM T78656 C7O5UG 11003379 Ki = 19 nM T78656 CJS79L 11011968 Ki = 9.8 nM T78656 CFB91X 11013959 Ki = 25 nM T78656 CSU4T7 11024618 Ki = 67 nM T78656 CX73TF 11035452 Ki = 12 nM T78656 C7ID8S 11043914 Ki = 210 nM T78656 CE0D8X 11044798 Ki = 6.9 nM T78656 C3G0FH 11046087 Ki = 7.4 nM T78656 CG0J7X 11047115 Ki = 42 nM T78656 C5N9GT 11056946 Ki = 7.1 nM T78656 C0FT4D 11067619 Ki = 7.3 nM T78656 CWK94J 11068036 Ki = 12 nM T78656 CL6Y9G 11068509 Ki = 16 nM T78656 C78OIE 11069268 Ki = 14 nM T78656 C0G3WS 11098166 Ki = 2.5 nM T78656 CH4UG6 11099817 Ki = 9.5 nM T78656 CK89UG 11101187 Ki = 7.5 nM T78656 CRU3M5 11110452 Ki = 6.3 nM T78656 C4VRT9 11111280 Ki = 20 nM T78656 CTBF50 11120893 Ki = 4.6 nM T78656 CDMI02 11121708 Ki = 19 nM T78656 CW6CZ1 11122117 Ki = 170 nM T78656 CV6RI1 11141562 Ki = 62 nM T78656 C9N5QU 11200511 Ki = 16 nM T78656 C6D1MZ 11223004 Ki = 12.3 nM T78656 C8OT1Q 11372635 Ki = 3.6 nM T78656 CBV52J 11384146 Ki = 2.7 nM T78656 CGX8F6 11596869 Ki > 2970000 nM T78656 C3T9XB 11727140 Ki = 11 nM T78656 CL97KG 11728004 Ki = 20 nM T78656 CYV02C 11747350 Ki = 2000 nM T78656 CG2WS6 11759467 Ki = 8.4 nM T78656 C0RTS1 11760896 Ki = 27 nM T78656 CQHI29 11808793 Ki = 3.8 nM T78656 CUI5G6 11809037 Ki = 4.7 nM T78656 CF9T0I 11810310 Ki = 11 nM T78656 CL1J7U 11822996 Ki = 19 nM T78656 C47SPL 11824009 Ki = 20 nM T78656 CVW4B5 11824522 Ki = 7.2 nM T78656 CHXQ26 18366015 IC50 = 363.08 nM T78656 CRU1N2 22611622 Ki = 9.7 nM T78656 C3HK0J 24865725 Ki = 501.19 nM T78656 C0O6FX 24865727 Ki = 1000 nM T78656 CI53SE 24893978 Ki = 7200 nM T78656 CPWJ26 44343212 Ki < 10000 nM T78656 CUXH48 44352308 EC50 = 6 nM T78656 CU1K6N 44352320 Ki = 1.6 nM T78656 CXO01L 44352344 Ki = 3.8 nM T78656 CQIA13 44386896 Ki = 2.9 nM T78656 CT6J0F 44387174 Ki = 3 nM T78656 CN02LY 44395762 Ki = 8.6 nM T78656 CLH1T7 44395786 Ki = 17 nM T78656 C9K4SC 44395787 Ki = 4.1 nM T78656 C93XHA 44395809 Ki = 4.8 nM T78656 CTA27N 44395810 Ki = 520 nM T78656 C9A4NM 44395832 Ki = 2.2 nM T78656 C52DPF 44395894 Ki = 12 nM T78656 CV86AM 44395925 Ki = 17 nM T78656 CVZ34J 44395930 Ki = 13 nM T78656 C4B0OI 44397588 Ki < 10000 nM T78656 C5FP0R 44397589 Ki < 1000 nM T78656 CE3G8U 44397670 Ki < 10000 nM T78656 CG0WO9 71459954 Ki = 17.8 nM T78656 CC6Q5R 72771081 Ki < 100 nM T78656 CAMF38 122190350 Ki = 8.3 nM T78656 C7LAR0 122190351 Ki = 1300 nM T78656 CW98LA 122190352 Ki = 41 nM T78656 C5CIU3 122190353 Ki = 530 nM T78656 C3BOY7 122190354 Ki = 1700 nM T78656 CPG19W 122190355 Ki = 870 nM T78656 CXR1O4 122190356 Ki = 610 nM T78656 CO21HS 122190357 Ki = 1100 nM T78656 CKP4A2 122190359 Ki = 3200 nM T78656 CZL80Q 122190360 Ki = 2400 nM T78656 D01HRV 9847194 IC50 > 10000 nM T78656 D03DET 10287730 Ki = 1995.26 nM T78656 D05XGR 6918647 Ki = 316.23 nM T78656 D07LRJ 5312149 Ki < 1000 nM T78656 D08CKM 9863250 Ki < 10000 nM T78656 D09PIN 3378093 Ki > 10000 nM T78656 D09WIL 10028436 Ki < 1995.26 nM T78656 D0F6CD 5202 EC50 = 7.9 nM T78656 D0H7PC 6918553 Ki > 10000 nM T78656 D0H9QG 5312148 Ki < 6309.57 nM T12475 D00RJJ 16130957 IC50 = 3.6 nM T12475 D01AHO 16131215 IC50 = 3.5 nM T12475 D04ODH 638793 IC50 = 10 nM T12475 D09OLZ 25074887 IC50 = 4.2 nM T12475 D0U5FF 657181 IC50 = 0.2884 nM T12475 D0VG7Y 24785956 Ki = 0.9 nM T12475 D0Y7KH 16136245 IC50 = 0.5754 nM T12475 D0F0UT 16137348 IC50 = 0.52 nM T12475 D0F2WP 10348973 IC50 = 0.08 nM T12475 D00VPV 3038517 IC50 = 0.06 nM T12475 D0D3ZP 11167850 Ki = 0.56 nM T12475 CV51AY 9807700 Ki = 11 nM T12475 CJ1E9O 9808288 IC50 = 0.7 nM T12475 CL0P7X 9809065 Ki = 1.2 nM T12475 C8NQ9Z 9809382 IC50 = 0.5 nM T12475 C50BTA 9809394 IC50 = 7.9 nM T12475 CWH9B0 9809590 IC50 = 0.2 nM T12475 CZ96QW 9823968 Ki = 83 nM T12475 C51SND 9825757 Ki = 250 nM T12475 CMEH32 9828154 Ki = 4200 nM T12475 C68VAU 9828888 IC50 = 0.5 nM T12475 C2VO4G 9829468 Ki = 5.2 nM T12475 C7UW8K 9831160 Ki = 2.7 nM T12475 CVF62U 9831689 IC50 = 0.2 nM T12475 C8LGT3 9850211 Ki = 30 nM T12475 C7U3GW 9851194 Ki = 1800 nM T12475 CV2DA6 9852184 Ki = 9 nM T12475 CPX6M4 9853275 IC50 = 0.2 nM T12475 CMDF10 9854500 Ki = 1.862 nM T12475 CQ4LC2 9872676 Ki = 0.4 nM T12475 C1TAK3 9873212 IC50 = 0.4 nM T12475 C8TSH7 9873394 IC50 = 300 nM T12475 C8GZI7 9873729 Ki = 42 nM T12475 CG2MY6 9875078 IC50 = 0.2 nM T12475 CDUK06 9891852 Ki = 16 nM T12475 CQT8A0 9892420 Ki = 34 nM T12475 C0W3DE 9893269 IC50 = 0.6 nM T12475 CFZ27W 9894997 IC50 = 0.3 nM T12475 C8EZ6R 9895596 IC50 = 0.3 nM T12475 CC4N2R 9895731 IC50 = 0.4 nM T12475 CSP3D6 9896373 IC50 = 0.3 nM T12475 CZT15H 9896737 IC50 = 0.6 nM T12475 CLYQ70 9910626 Ki = 56 nM T12475 C1U0WA 9911446 Ki = 17 nM T12475 C4IW7L 9915597 Ki = 72 nM T12475 C3H4TW 9916573 Ki = 500 nM T12475 CG8F3V 9917213 IC50 = 30 nM T12475 CA4Q9C 9917618 IC50 = 0.4 nM T12475 CW7NQ2 9918188 IC50 = 3 nM T12475 CZY34G 9938925 IC50 = 0.4 nM T12475 CYM57O 9939030 Ki = 50 nM T12475 CB2T5O 9939837 IC50 = 0.1 nM T12475 C1ZUF7 9958318 IC50 = 16 nM T12475 CVB2K6 9959327 Ki = 160 nM T12475 C41ZOX 9960268 Ki = 59 nM T12475 C4N8ED 9960399 IC50 = 2.8 nM T12475 CM0XL1 9961721 IC50 = 0.31 nM T12475 C2U0ZV 9979079 IC50 = 357 nM T12475 CJE42Z 9983568 Ki = 4.1 nM T12475 C2DM0Q 9984259 Ki = 8.1 nM T12475 CTG8J9 9985901 IC50 = 0.3 nM T12475 C2M0EZ 9986320 Ki = 4.6 nM T12475 CJYD27 10007333 Ki = 20 nM T12475 C1F2RH 10008768 IC50 = 0.3 nM T12475 CWV42E 10009345 IC50 = 0.3 nM T12475 C3DKJ8 10027591 Ki = 3 nM T12475 C2A1HR 10032222 IC50 = 6.4 nM T12475 CZ54AR 10050123 Ki = 13 nM T12475 CF6KG7 10051739 Ki = 4.5 nM T12475 C70LEU 10053165 IC50 = 0.3 nM T12475 C3L4WH 10074296 IC50 = 7 nM T12475 CEJK75 10077523 IC50 = 2 nM T12475 CJ0DZ1 10077844 Ki = 2.8 nM T12475 CO1CJ8 10098618 Ki = 20 nM T12475 CVHC47 10100930 IC50 = 0.07 nM T12475 CA46SM 10187208 IC50 = 0.6 nM T12475 C0L7JD 10208964 IC50 = 243 nM T12475 CIQ16S 10226423 Ki = 110 nM T12475 CZ9R4X 10258658 IC50 = 3.2 nM T12475 CI5CH2 10311600 Ki = 1 nM T12475 CT3P8Q 10323198 Ki = 2 nM T12475 C2YN9G 10345138 Ki = 0.61 nM T12475 C93URC 10347081 Ki = 20 nM T12475 C61PRI 10371708 IC50 = 0.12 nM T12475 C3JIZ5 10394119 Ki = 9.3 nM T12475 C7BRW4 10438167 IC50 = 15 nM T12475 CUJB47 10439419 Ki = 7.5 nM T12475 CNI16O 10439527 Ki = 25 nM T12475 CX2V8Z 10603202 IC50 = 4 nM T12475 CWV38O 10624976 IC50 = 2000 nM T12475 CH19LT 10649568 Ki = 0.4 nM T12475 CX0QW2 10674894 IC50 = 6 nM T12475 CV34AE 10722009 IC50 = 70 nM T12475 CJ2Y9O 10794239 IC50 = 0.2 nM T12475 CDRE17 10837806 IC50 = 10000 nM T12475 CW0JF2 10874838 Ki = 1700 nM T12475 CG5DN6 10875519 Ki = 7700 nM T12475 C9PFN4 10886383 Ki = 30 nM T12475 C60MWX 10897903 IC50 = 20 nM T12475 C8YZ6N 10907714 Ki = 4800 nM T12475 C48IRB 10908122 Ki = 400 nM T12475 CT6E8S 10919052 Ki = 36 nM T12475 CIOC73 10919567 IC50 = 0.4 nM T12475 C89ILX 10929574 Ki = 240 nM T12475 C8E0VN 10929667 Ki = 24 nM T12475 C82SJD 10929801 Ki = 300 nM T12475 C3E1PG 10930118 Ki = 130 nM T12475 CJA61E 10930638 IC50 = 13 nM T12475 CR1WT2 10940289 Ki = 230 nM T12475 CMC1B7 10951713 Ki = 130 nM T12475 CEAV16 10962804 Ki = 190 nM T12475 C6P0OV 10983979 Ki = 1100 nM T12475 CZ2A7G 10983989 Ki = 480 nM T12475 C1F5XB 10985312 IC50 = 0.3 nM T12475 CA3QK1 10994908 Ki = 220 nM T12475 CJ6OU9 10995320 Ki = 320 nM T12475 CB61IC 10995569 Ki = 4.2 nM T12475 CGAO93 11005990 Ki = 38 nM T12475 C8ZSR6 11017929 IC50 = 1 nM T12475 CJ8DM4 11027376 Ki = 400 nM T12475 CVQP20 11049737 Ki = 530 nM T12475 CRMV80 11050145 Ki = 7.9 nM T12475 CW57YC 11050500 Ki = 5100 nM T12475 C1QHU6 11071561 Ki = 2200 nM T12475 CZLG13 11082604 Ki = 9200 nM T12475 C38QUM 11092567 Ki = 430 nM T12475 C0SR5E 11103551 Ki = 430 nM T12475 CF6M8B 11103767 Ki = 8 nM T12475 CZ58OK 11113778 Ki = 3800 nM T12475 CG1Y8H 11123821 Ki = 240 nM T12475 CH9O5M 11124671 Ki = 4800 nM T12475 CTV0P2 11124921 Ki = 490 nM T12475 CJTI91 11137010 IC50 = 10.5 nM T12475 CPS20T 11145953 Ki = 350 nM T12475 CZM5D1 11156980 Ki = 5.6 nM T12475 CRYB13 11157017 Ki = 700 nM T12475 CE9T2V 11168176 Ki = 1200 nM T12475 CLH40V 11168311 Ki = 2.8 nM T12475 CV18TH 11168330 Ki = 400 nM T12475 C9HUM0 11168634 Ki = 120 nM T12475 C2IAS0 11168776 Ki = 1.8 nM T12475 CFV67S 11178994 Ki = 39 nM T12475 CO3N9K 11179420 Ki = 13 nM T12475 CXU0S9 11179660 Ki = 130 nM T12475 CQ6U1C 11179922 Ki = 70 nM T12475 C5N9YL 11180219 Ki = 6.5 nM T12475 C1YNA4 11191153 Ki = 22 nM T12475 CHKZ83 11191674 Ki = 5 nM T12475 CM34TB 11191675 Ki = 3.6 nM T12475 CQ0Z6C 11192019 Ki = 66 nM T12475 CKXI78 11192229 Ki = 15 nM T12475 CQHW25 11202636 Ki = 1.2 nM T12475 CMIA32 11202795 Ki = 51 nM T12475 CCVO71 11214294 Ki = 5.1 nM T12475 C4SHP0 11214295 Ki = 75 nM T12475 CAL67V 11214614 Ki = 4.5 nM T12475 CQA03J 11214860 Ki = 15 nM T12475 C08LHX 11225384 Ki = 37 nM T12475 CH52BG 11225960 Ki = 16 nM T12475 C0NZG6 11226171 Ki = 79 nM T12475 CD2X4S 11226470 Ki = 3 nM T12475 COX1Y7 11226531 Ki = 4 nM T12475 CGP1U9 11226753 Ki = 6.5 nM T12475 C5PUZ6 11226884 IC50 = 400 nM T12475 CIF71C 11227010 Ki = 10800 nM T12475 C5PSE2 11236870 Ki = 6.4 nM T12475 C13FWV 11237922 IC50 = 120 nM T12475 CS6N3H 11238091 Ki = 64 nM T12475 C0PQ1H 11238459 Ki = 470 nM T12475 CWYJ92 11238637 Ki = 200 nM T12475 C7MVO9 11249167 Ki = 15 nM T12475 CT43KJ 11249548 IC50 = 6.1 nM T12475 C9SP6Z 11260648 Ki = 370 nM T12475 CV8XS1 11260704 Ki = 81 nM T12475 CXAD47 11261195 Ki = 46 nM T12475 C15QDU 11261693 Ki = 14 nM T12475 CD7J9T 11262242 IC50 = 0.6 nM T12475 CFQB10 11272935 Ki = 20 nM T12475 CH5X4I 11282957 Ki = 2.3 nM T12475 CTO36S 11283517 Ki = 140 nM T12475 C4E2IA 11283954 Ki = 4.1 nM T12475 C5JLA6 11284264 Ki = 4800 nM T12475 CHZG95 11284357 Ki = 880 nM T12475 CZJ1X4 11294757 Ki = 1100 nM T12475 CFN37P 11294792 Ki = 6.4 nM T12475 CH83MP 11294949 Ki = 970 nM T12475 CP0W4R 11295556 Ki = 680 nM T12475 CVKX03 11307227 Ki = 8.5 nM T12475 C27VMA 11318370 Ki = 18 nM T12475 CRC62Z 11318649 IC50 = 750 nM T12475 CC65PV 11319401 Ki = 27 nM T12475 CO8AF2 11319703 Ki = 180 nM T12475 CN36IG 11329628 Ki = 880 nM T12475 CN4C2X 11330034 Ki = 110 nM T12475 C8RNH1 11330072 Ki = 1500 nM T12475 CT3NA8 11330164 IC50 = 160 nM T12475 C4CK8B 11330280 Ki = 140 nM T12475 CNH18O 11330603 Ki = 100 nM T12475 C74LWO 11331001 Ki = 1.2 nM T12475 C9PW4N 11341364 Ki = 13 nM T12475 CL83BG 11341990 Ki = 63 nM T12475 CTC0V6 11352630 Ki = 220 nM T12475 CD6LJ2 11352834 Ki = 340 nM T12475 CT37AI 11353175 Ki = 7 nM T12475 C4KZH9 11354193 Ki = 21 nM T12475 CGN21Z 11363829 Ki = 71 nM T12475 CSZD83 11364940 Ki = 0.2 nM T12475 CT6MO8 11365653 Ki = 1 nM T12475 C0FYS9 11374717 Ki = 5.6 nM T12475 CAY34E 11375759 Ki = 3.1 nM T12475 C5UJC8 11375912 Ki = 370 nM T12475 CY8O2J 11376064 Ki = 1400 nM T12475 C6C3BF 11376252 Ki = 0.45 nM T12475 CIHS32 11386605 Ki = 460 nM T12475 CP85KM 11387100 Ki = 7.9 nM T12475 C74MPZ 11421243 Ki = 240 nM T12475 C89KJA 11421385 Ki = 53 nM T12475 CSU47B 11421412 IC50 = 0.5 nM T12475 CY74AZ 11421518 Ki = 3.7 nM T12475 C3VR2T 11431754 Ki = 94 nM T12475 CHW53K 11443571 Ki = 1200 nM T12475 C37RYL 11443711 Ki = 0.6 nM T12475 C0XD7Y 11444384 Ki = 61 nM T12475 CL5V0D 11444885 Ki = 4 nM T12475 CV19KF 11444886 Ki = 3.1 nM T12475 C9W3SM 11455176 Ki = 780 nM T12475 CW96YL 11455317 Ki = 3.4 nM T12475 C5CGK7 11456285 Ki = 3.6 nM T12475 CN3AX6 11461935 Ki > 100000 nM T12475 CZP21R 11466452 Ki = 2.4 nM T12475 C4GX9F 11467134 Ki = 19 nM T12475 CU7S8C 11467328 Ki = 170 nM T12475 CDZ53U 11467552 Ki = 3.162 nM T12475 C2N3EZ 11477615 Ki = 7.5 nM T12475 C7CYI9 11477970 Ki = 25 nM T12475 CQ19VY 11477988 IC50 = 0.5 nM T12475 C38OME 11478448 IC50 < 10 nM T12475 CB9N7C 11489334 Ki = 965 nM T12475 CC7D9K 11490288 Ki = 21 nM T12475 CX0J2W 11490509 Ki = 4.6 nM T12475 CV3H7G 11496945 IC50 = 14 nM T12475 CLIN17 11511860 IC50 = 5000 nM T12475 C9PDV4 11512807 IC50 = 7000 nM T12475 CY8M0L 11512905 IC50 = 0.1 nM T12475 CU79WP 11518185 IC50 = 38 nM T12475 CT3VE0 11520078 IC50 = 100 nM T12475 C8CRV4 11525358 IC50 = 7 nM T12475 C5NG9E 11525693 IC50 = 18 nM T12475 CX3B0G 11526254 IC50 = 5.2 nM T12475 CQ2EW1 11527301 IC50 = 300 nM T12475 C7YN0P 11527384 IC50 = 400 nM T12475 C06COY 11532637 IC50 = 6.7 nM T12475 CFQ5X6 11549071 IC50 = 9 nM T12475 CYL4F1 11563584 IC50 = 0.06 nM T12475 CNE60T 11570616 IC50 = 500 nM T12475 CDA01M 11583388 IC50 = 58 nM T12475 COM54B 11583756 Ki = 12.2 nM T12475 CE0G4Q 11592473 IC50 = 2000 nM T12475 CAU32N 11592658 IC50 = 8 nM T12475 C9AXV6 11592777 IC50 = 0.4 nM T12475 CN6LS5 11599857 IC50 = 100 nM T12475 CKV14Z 11604354 IC50 = 7.5 nM T12475 CNA39D 11606766 IC50 = 200 nM T12475 CH0MI9 11614283 IC50 = 0.4 nM T12475 CI5J4K 11618517 IC50 = 21 nM T12475 CT0A3I 11619461 IC50 = 22 nM T12475 C2HC3R 11619584 IC50 > 20000 nM T12475 C9FL0O 11619758 IC50 = 11000 nM T12475 C13YEW 11620431 IC50 = 9.7 nM T12475 CAE5L7 11626096 IC50 = 33 nM T12475 CM1W6Y 11628915 IC50 = 0.2 nM T12475 CTXR53 11634198 IC50 = 18 nM T12475 CLW74P 11635837 IC50 = 300 nM T12475 CQK1U0 11642933 IC50 = 30 nM T12475 C6Z2DO 11643195 IC50 = 0.2 nM T12475 C19DQJ 11671279 Ki = 2 nM T12475 C7HQ2Y 11692806 IC50 = 200 nM T12475 C6Z9GJ 11692959 IC50 = 0.07 nM T12475 CP9Z1E 11700433 IC50 = 0.1 nM T12475 C58JXM 11707186 IC50 = 0.1 nM T12475 COV9F5 11712618 IC50 = 21 nM T12475 C5G1BP 11720984 IC50 = 170 nM T12475 CM8NK4 11733484 Ki = 1700 nM T12475 C0DMC4 11751752 Ki = 595 nM T12475 CJ0T5N 11752130 Ki = 10 nM T12475 CQ7C2S 11752557 Ki = 500 nM T12475 CUO6C9 11763365 Ki = 12000 nM T12475 CNB97I 11766904 Ki = 260 nM T12475 C2JR5X 11785958 Ki = 320 nM T12475 CN28CA 11786039 Ki = 460 nM T12475 CQB2S7 11999836 IC50 > 10000 nM T12475 CST2O1 11999838 IC50 > 10000 nM T12475 C6QP0V 12094521 Ki > 10000 nM T12475 C4QOA5 12986401 Ki = 110 nM T12475 CH58CX 12991507 Ki = 230 nM T12475 CU0I1H 15462657 IC50 = 50 nM T12475 C4BD9W 15462660 IC50 = 400 nM T12475 CX5A9K 15462663 IC50 = 30 nM T12475 C1KI6H 15462665 IC50 = 700 nM T12475 CJ5OZ8 15462666 Ki = 180 nM T12475 C90NVW 15602804 IC50 = 20 nM T12475 CZES74 15602805 IC50 = 2.3 nM T12475 C9D8SX 15602806 IC50 = 9.8 nM T12475 CN0TK4 15602807 IC50 = 47 nM T12475 CE84FR 15602808 IC50 = 39 nM T12475 CB4WA3 15604462 IC50 > 10000 nM T12475 CLQ91O 16058727 Ki = 2.3 nM T12475 CWJ97K 16144222 IC50 = 8.6 nM T12475 CZY14F 16144515 IC50 = 6.1 nM T12475 C0RM9G 16144824 IC50 = 7.8 nM T12475 CBD65G 16144832 IC50 = 7.2 nM T12475 C37EZO 16144863 IC50 = 9.5 nM T12475 CR04QN 16144865 IC50 = 8.9 nM T12475 CQD3X6 16145403 IC50 = 5 nM T12475 C20JCU 16146016 IC50 = 10.8 nM T12475 CX1M8P 16146022 IC50 = 3 nM T12475 CS8Q5Y 16146554 IC50 = 5.5 nM T12475 CEGQ10 16146884 IC50 = 9.1 nM T12475 CL9B7E 16147451 IC50 = 8.1 nM T12475 CI0S3O 16147453 IC50 = 5.6 nM T12475 CDL18K 16147757 IC50 = 7.7 nM T12475 CD3ZF2 16147767 IC50 = 4.3 nM T12475 C28TLC 16148338 IC50 = 7 nM T12475 CXG07F 16155157 IC50 = 1.37 nM T12475 C9AI1F 16155285 IC50 = 2.951 nM T12475 CV97DN 16155294 IC50 = 2.04 nM T12475 CYN7P0 16155358 IC50 = 1.61 nM T12475 CO54BM 16155412 IC50 = 4.55 nM T12475 C7UOF3 16156049 IC50 = 2.13 nM T12475 CNKP47 16156105 IC50 = 2.951 nM T12475 CCA36D 16156328 IC50 = 1.479 nM T12475 CU5PJ8 16156341 IC50 = 1.66 nM T12475 C1PW8V 16156572 IC50 = 4.99 nM T12475 C3KZJ1 16156638 IC50 = 1.479 nM T12475 CYTL52 16156639 IC50 = 4.169 nM T12475 C2R6KJ 16156643 IC50 = 1.12 nM T12475 CW2I3V 16156649 IC50 = 2.55 nM T12475 C4K9UL 16156706 IC50 = 9.55 nM T12475 CG48LX 16157293 IC50 = 2.8 nM T12475 CPK4E3 17757565 Ki = 5 nM T12475 C58CJL 17757566 Ki = 5 nM T12475 CD08XF 18324807 IC50 = 0.08 nM T12475 CP72XJ 20691661 IC50 = 0.1 nM T12475 C7C4GB 20728209 Ki = 700 nM T12475 CW3VX1 21018389 Ki = 1.1 nM T12475 CJX3M8 21036877 Ki = 1.1 nM T12475 C57CRP 21036878 Ki = 1.2 nM T12475 C09MOY 21045797 Ki = 20 nM T12475 CKQT59 21045805 Ki = 33 nM T12475 CDGU29 21045807 Ki = 780 nM T12475 CJI5Z9 21045817 Ki = 67 nM T12475 C6OEN5 21045818 Ki = 130 nM T12475 CK0S9D 21045823 Ki = 66 nM T12475 C71UKR 21045828 Ki = 74 nM T12475 C6S8TJ 21045829 Ki = 40 nM T12475 C6U4ZX 21045831 Ki = 700 nM T12475 C7LY4W 21045833 Ki = 150 nM T12475 CRU51H 21045834 Ki = 110 nM T12475 CZVG59 21046387 Ki = 51 nM T12475 C0WM6V 21046569 Ki = 510 nM T12475 C38OVD 21046570 Ki = 24 nM T12475 CJS06P 21046762 Ki = 220 nM T12475 C3I6AO 21047516 Ki = 44 nM T12475 CB7Y9X 21047518 Ki = 35 nM T12475 CP1AO0 21047519 Ki = 29 nM T12475 CTA7S8 21047534 Ki = 11 nM T12475 CZ2JG5 21047538 Ki = 220 nM T12475 C2QS6H 21047583 Ki = 80 nM T12475 C8E7CT 21047618 Ki = 14 nM T12475 CC63KH 21047631 Ki = 174 nM T12475 C2RPI6 21047633 Ki = 91 nM T12475 C50PMJ 21047784 Ki = 24 nM T12475 CHSM29 21047785 Ki = 103 nM T12475 C8DL4W 21047799 Ki = 180 nM T12475 CJ2AC6 21047805 Ki = 300 nM T12475 C2RO7V 21047807 Ki = 63 nM T12475 CM56VB 21047815 Ki = 170 nM T12475 C0Q4DJ 21047858 Ki = 42 nM T12475 CGP48D 21047859 Ki = 140 nM T12475 CT51QF 21047937 Ki = 79 nM T12475 C3FT2H 21048269 Ki = 102 nM T12475 C16QAR 21048323 Ki = 180 nM T12475 C8LHG6 21048462 Ki = 54 nM T12475 C7PK5R 21355220 Ki = 6 nM T12475 CW8M5K 21899433 IC50 = 162 nM T12475 CGD56N 22100905 IC50 = 58 nM T12475 C5OP6A 22716524 Ki = 230 nM T12475 CKMI15 22716552 Ki = 40 nM T12475 CAW8J4 22716564 Ki = 220 nM T12475 CM35YS 22716581 Ki = 4.5 nM T12475 C0MKD9 22716607 Ki = 93 nM T12475 C5BZ7K 23450008 Ki = 120 nM T12475 C36YOW 23656390 IC50 = 1.5 nM T12475 CAK10D 24825725 IC50 = 5.8 nM T12475 CY6JX9 24857895 Ki = 33 nM T12475 CZC3U8 25113693 Ki = 140 nM T12475 CWC26X 25156399 Ki = 71 nM T12475 CNOJ07 25156400 Ki = 2.1 nM T12475 C5Z1RT 25156669 Ki = 7.6 nM T12475 CQY6Z1 25156942 Ki = 3.7 nM T12475 CUE0Z5 25156943 Ki = 1.1 nM T12475 CQ6PI5 25156944 Ki = 4.2 nM T12475 C5ZJX4 25156946 Ki = 12 nM T12475 CIK26N 25193700 IC50 = 220 nM T12475 CED7L6 25193797 IC50 = 120 nM T12475 CT5ZM7 25193798 IC50 = 1200 nM T12475 CDQ9N2 25194090 IC50 = 1300 nM T12475 CJT2O8 25194091 IC50 = 120 nM T12475 CCF94J 25194092 IC50 = 1200 nM T12475 C4P2KV 44185958 IC50 = 89 nM T12475 CRM98S 44215053 IC50 = 14 nM T12475 CSR1G3 44215055 IC50 = 18 nM T12475 C39VFI 44215908 IC50 = 381 nM T12475 CPSK12 44215933 Ki = 6 nM T12475 CW8T9L 44267810 Ki = 22.39 nM T12475 CNP72I 44267811 Ki = 2041.74 nM T12475 CV97XW 44267812 Ki = 15.14 nM T12475 C9S3IO 44267863 Ki = 275.42 nM T12475 CWJ57P 44267864 Ki = 562.34 nM T12475 CEX30Z 44267865 Ki = 66.07 nM T12475 CA0Y7T 44267866 Ki = 36.31 nM T12475 C5ANG7 44267868 Ki = 3.89 nM T12475 CT9OJ0 44267869 Ki < 100 nM T12475 C62ZFA 44267870 Ki = 79.43 nM T12475 C1RF7E 44267874 Ki = 213.8 nM T12475 CC6L2T 44267875 Ki = 51.29 nM T12475 C4YPM6 44267876 Ki = 114.82 nM T12475 CP6VC9 44267881 Ki = 1621.81 nM T12475 CMX53U 44267882 Ki = 630.96 nM T12475 CT0S9X 44267883 Ki = 10000 nM T12475 CY3JD1 44267885 Ki = 2041.74 nM T12475 CP7HY6 44267887 Ki = 5.623 nM T12475 C8WC3G 44267902 Ki = 18.62 nM T12475 CQ8M1C 44267903 Ki = 4677.35 nM T12475 C1SCA4 44267904 Ki = 794.33 nM T12475 CDE3O8 44267905 Ki = 5623.41 nM T12475 CE2YU5 44267906 Ki = 48.98 nM T12475 C4RU6L 44267907 Ki = 0.3311 nM T12475 CGJ13K 44274227 IC50 = 20 nM T12475 C9GKY5 44274228 IC50 = 200 nM T12475 C94YST 44274229 IC50 = 200 nM T12475 C92DFY 44274247 IC50 = 20 nM T12475 C5LH1J 44274248 IC50 = 80 nM T12475 CE28CD 44274327 IC50 = 400 nM T12475 CN9CU3 44274475 IC50 = 200 nM T12475 CVY7J6 44287759 Ki = 1.514 nM T12475 CNQ4S7 44287778 Ki = 27.54 nM T12475 C2N9ML 44287779 Ki = 204.17 nM T12475 C74SJK 44287893 Ki = 18.62 nM T12475 C8Z7PR 44288073 Ki = 7.586 nM T12475 CE8SY2 44288074 Ki = 13.18 nM T12475 C4XHQ7 44288075 Ki ~ 5 nM T12475 C8L3VH 44288078 Ki = 190.55 nM T12475 C0JVW3 44288079 Ki = 79.43 nM T12475 C5OI0D 44288080 Ki = 0.8511 nM T12475 CHW6B1 44288081 Ki = 1.288 nM T12475 CO8T2I 44288082 Ki = 7.244 nM T12475 CAMG30 44292868 IC50 = 1.1 nM T12475 C3QXV0 44292869 IC50 = 2 nM T12475 CJ27QW 44292918 IC50 = 7.1 nM T12475 CYPO82 44292919 IC50 = 5 nM T12475 C5FYT9 44292939 IC50 = 2.3 nM T12475 C1B6AY 44292950 IC50 = 1.1 nM T12475 C1PL2M 44293045 IC50 = 0.7 nM T12475 C3ATD8 44293081 IC50 = 1.8 nM T12475 C3MGW9 44293111 IC50 = 10 nM T12475 CXT4Q8 44293130 IC50 = 32 nM T12475 CWR5Q3 44293131 IC50 = 32 nM T12475 CAJ10V 44293134 IC50 = 36 nM T12475 CQS13K 44293151 IC50 = 11 nM T12475 CE6W4S 44293164 IC50 = 55 nM T12475 CUJC52 44293165 IC50 = 45 nM T12475 CJ1OI8 44293205 IC50 = 0.5 nM T12475 CZWP67 44293206 IC50 = 0.7 nM T12475 CJO7Q8 44293222 IC50 = 0.9 nM T12475 CF1WG5 44293249 IC50 = 18 nM T12475 CSR7N6 44293250 IC50 = 59 nM T12475 CBL34G 44293274 IC50 = 58 nM T12475 CP74KZ 44293284 IC50 = 3.9 nM T12475 C1ZT9C 44293285 IC50 = 57 nM T12475 CI4U2C 44293305 IC50 = 61 nM T12475 CNX1A4 44293335 IC50 = 22 nM T12475 CDH8Q7 44293347 IC50 = 62 nM T12475 CA5NQ9 44293348 IC50 = 2.3 nM T12475 CZ46XW 44293376 IC50 = 40 nM T12475 CC3Q5Y 44293377 IC50 = 38 nM T12475 CHDW46 44293378 IC50 = 300 nM T12475 CC83OZ 44293386 IC50 = 1 nM T12475 C7EY9U 44293484 IC50 = 200 nM T12475 CK8W1G 44293485 IC50 = 90 nM T12475 C9GOI6 44293486 IC50 = 54 nM T12475 CXFH09 44293487 IC50 = 8.3 nM T12475 CW2C3E 44293488 IC50 = 22 nM T12475 CY40TU 44293511 IC50 = 94 nM T12475 CW6P1S 44293555 IC50 = 170 nM T12475 CFJC54 44293591 IC50 = 12 nM T12475 CZD2O3 44293592 IC50 = 190 nM T12475 C17AUE 44293594 IC50 = 260 nM T12475 CZGI52 44293617 IC50 = 3.6 nM T12475 CG2O7D 44293802 IC50 = 38 nM T12475 CBTJ83 44293803 IC50 = 15 nM T12475 CN6D2E 44295109 Ki = 6400 nM T12475 CS6Q5R 44295630 IC50 = 5.7 nM T12475 CNM6P8 44295699 IC50 = 0.5 nM T12475 C7NHT2 44295753 IC50 = 0.6 nM T12475 CNK73E 44295755 IC50 = 0.9 nM T12475 CS52RI 44296258 IC50 = 2 nM T12475 CG2SE4 44305274 IC50 = 7 nM T12475 CPYJ37 44305285 IC50 = 0.7 nM T12475 CVK7N8 44305286 IC50 = 3 nM T12475 C1L9IK 44305306 IC50 = 20 nM T12475 CW9S2I 44305362 IC50 = 3 nM T12475 C7V1DY 44305604 IC50 = 5 nM T12475 CJ2KZ4 44305605 IC50 = 10 nM T12475 CG4WU2 44309252 Ki = 2500 nM T12475 C4DK5J 44309296 Ki = 150 nM T12475 CU63TQ 44309319 Ki = 80 nM T12475 C3G5HF 44309321 Ki = 220 nM T12475 C3E1ZQ 44309323 Ki = 2200 nM T12475 C15UTE 44309357 Ki = 41 nM T12475 CJWP52 44309359 Ki = 56 nM T12475 C7LEV2 44309361 Ki = 28000 nM T12475 C0T2PY 44309372 Ki = 370 nM T12475 C8H5NY 44309375 Ki = 290 nM T12475 C14CFL 44309376 Ki = 300 nM T12475 CSD60N 44309388 Ki = 9500 nM T12475 CG6UV8 44309390 Ki = 18 nM T12475 C54WNT 44309399 Ki = 28000 nM T12475 C9MW6U 44309403 Ki = 1400 nM T12475 CXS20N 44309404 Ki = 67 nM T12475 C6YMK5 44309439 Ki = 110 nM T12475 C4QK8N 44309440 Ki = 11 nM T12475 C9K2NU 44309511 Ki = 12 nM T12475 CLN41T 44309522 Ki = 30000 nM T12475 C70UEG 44309525 Ki = 230 nM T12475 CS17NK 44309535 Ki = 14 nM T12475 CY12EH 44309541 Ki = 110 nM T12475 C30TJM 44309559 Ki = 47 nM T12475 CH57IZ 44309572 IC50 = 0.44 nM T12475 CU19GP 44309573 Ki = 130 nM T12475 CJ8ZP2 44309576 Ki = 36 nM T12475 C06OJI 44309582 Ki = 230 nM T12475 C86ENC 44309585 Ki = 29 nM T12475 CO9DA7 44309615 Ki = 100 nM T12475 CNR9V8 44309616 Ki = 140 nM T12475 C6CDU8 44309617 Ki = 79 nM T12475 C0SZV8 44309631 Ki = 52 nM T12475 C8DBA3 44309652 Ki = 65 nM T12475 C25PSZ 44309671 Ki = 950 nM T12475 CC2Y3G 44312664 Ki > 10000 nM T12475 CZM1B8 44312666 Ki = 260 nM T12475 CH3NV1 44312724 Ki = 140 nM T12475 C74KJT 44312779 Ki > 10000 nM T12475 CMQ6T7 44312806 Ki = 430 nM T12475 CDA3K8 44312821 Ki = 230 nM T12475 C0F6HJ 44313011 Ki > 10000 nM T12475 CK03YH 44313105 Ki > 10000 nM T12475 C7QVS6 44320895 IC50 = 2.6 nM T12475 C6X8FN 44320921 IC50 = 1.2 nM T12475 C2R0KY 44321052 IC50 = 0.3 nM T12475 C0UC7O 44321100 IC50 = 2.1 nM T12475 CI10XM 44321101 IC50 = 1 nM T12475 C2B4AM 44321146 IC50 = 39 nM T12475 CO83ML 44321147 IC50 = 2.7 nM T12475 CAE18S 44321148 IC50 = 0.6 nM T12475 CNZ2T7 44321290 IC50 = 0.8 nM T12475 C4ODM3 44321291 IC50 = 4.8 nM T12475 CQB87O 44321292 IC50 = 6.8 nM T12475 CP0ZN4 44321345 IC50 = 8.2 nM T12475 CB73WQ 44321393 IC50 = 0.6 nM T12475 C68QFC 44321394 IC50 = 11 nM T12475 COKZ03 44321410 IC50 = 1 nM T12475 C0DG3L 44321411 IC50 = 0.4 nM T12475 C9I7XO 44321412 IC50 = 8.8 nM T12475 CI6HX8 44321458 IC50 = 21 nM T12475 CJ4K8W 44321496 IC50 = 4.4 nM T12475 C18PDZ 44321497 IC50 = 6.1 nM T12475 C5L4NO 44321498 IC50 = 0.7 nM T12475 CFH60J 44321509 IC50 = 1.4 nM T12475 CF5QV6 44321510 IC50 = 5.6 nM T12475 CZ4UA9 44321695 IC50 = 82 nM T12475 C3WJU9 44321963 IC50 = 0.4 nM T12475 CY5CQ2 44321964 IC50 = 1.4 nM T12475 CS34KT 44340612 Ki = 550 nM T12475 CNFX74 44340623 Ki = 90 nM T12475 CV94JR 44340631 Ki = 1200 nM T12475 CK4D2W 44340632 Ki = 430 nM T12475 CB4W1H 44340635 Ki = 190 nM T12475 C5SF8Z 44340636 Ki = 2500 nM T12475 CKNG30 44340637 Ki = 5 nM T12475 CE8JX7 44340641 Ki = 81 nM T12475 CA5US9 44340642 Ki = 950 nM T12475 COZ92E 44340643 Ki = 8300 nM T12475 CDTZ17 44340644 Ki = 280 nM T12475 C6SCB9 44340646 Ki = 53 nM T12475 CAZ5D1 44340649 Ki = 18000 nM T12475 CR1ZC8 44340652 Ki = 5 nM T12475 CZ7Q0K 44340656 Ki = 470 nM T12475 CMJV54 44340670 Ki = 2000 nM T12475 CCWX09 44340688 Ki = 96 nM T12475 C27UKF 44340697 Ki = 550 nM T12475 CG76VD 44340720 Ki = 150 nM T12475 C3INX6 44340749 Ki = 1.1 nM T12475 CLW19C 44340771 Ki = 330 nM T12475 C4TU3E 44340780 Ki = 240 nM T12475 C05OLF 44340783 Ki = 210 nM T12475 C4KFS8 44340784 Ki = 250 nM T12475 CHB56J 44340785 Ki = 170 nM T12475 CZ6F8G 44340788 Ki = 12 nM T12475 CP5WX1 44340798 Ki = 280 nM T12475 CO1JZ9 44340804 Ki = 250 nM T12475 CQ4OX8 44340808 Ki = 32 nM T12475 CYXN72 44340824 Ki = 85 nM T12475 CI91SE 44340825 Ki = 310 nM T12475 CS4I8Y 44340840 Ki = 720 nM T12475 CQF5N1 44340844 Ki = 590 nM T12475 C1ZF9T 44340845 Ki = 1600 nM T12475 CXH0Y1 44340860 Ki = 7000 nM T12475 C16WPU 44340888 IC50 = 0.4 nM T12475 CJPO47 44340906 IC50 = 0.3 nM T12475 CQS6A9 44340928 IC50 = 20 nM T12475 CX56ZP 44340929 IC50 = 0.6 nM T12475 C9SO6I 44341046 IC50 = 0.4 nM T12475 CMA19W 44341056 IC50 = 0.8 nM T12475 C72XIY 44341057 Ki = 1800 nM T12475 C8HJF1 44341074 Ki = 780 nM T12475 CU9JO4 44341075 Ki = 15000 nM T12475 C9CT6J 44341080 IC50 = 4.6 nM T12475 C2H4BC 44341081 IC50 = 19 nM T12475 C1BGQ9 44341082 IC50 = 0.4 nM T12475 C8T1WH 44341113 IC50 = 0.9 nM T12475 CF0YH8 44341164 IC50 = 0.8 nM T12475 CH69VI 44341186 IC50 = 8.2 nM T12475 C7JV8Q 44341197 IC50 = 0.7 nM T12475 CS68GY 44341198 IC50 = 0.7 nM T12475 CU09QW 44341199 IC50 = 0.9 nM T12475 CS5PG0 44343779 Ki = 12 nM T12475 C96DUZ 44343804 Ki = 12 nM T12475 CQ48GR 44343881 Ki = 92 nM T12475 CV27ET 44343914 Ki = 100 nM T12475 CI4UF3 44343931 Ki = 55 nM T12475 CZ9VC3 44343932 Ki = 24000 nM T12475 CQ84HZ 44343975 Ki = 200 nM T12475 C43CYT 44343976 Ki = 2600 nM T12475 CZC3M1 44344157 Ki = 23 nM T12475 CQZ25F 44346239 Ki = 58 nM T12475 CR19BA 44346260 Ki = 360 nM T12475 CPK54W 44346261 Ki = 150 nM T12475 C80KJQ 44346348 Ki = 43 nM T12475 CIAV19 44346349 Ki = 300 nM T12475 CO93UT 44346374 Ki = 270 nM T12475 CW29ZO 44346375 Ki = 16 nM T12475 CF1BY8 44346376 Ki = 11 nM T12475 C2FNX3 44346396 Ki = 9 nM T12475 CF1M3Q 44346397 Ki = 0.6 nM T12475 C90NLC 44346398 Ki = 170 nM T12475 C68QLC 44346479 Ki = 17 nM T12475 C4P5SO 44346594 Ki = 640 nM T12475 CZFA83 44346649 Ki = 460 nM T12475 CK48EO 44346662 Ki = 76 nM T12475 C2QD4X 44346663 Ki = 170 nM T12475 CM2AB8 44346665 Ki = 88 nM T12475 CZ0V8W 44346666 Ki = 61 nM T12475 CR7AE5 44346667 Ki = 4.1 nM T12475 CI0L2H 44346848 Ki = 175 nM T12475 CKP87A 44347004 Ki = 28 nM T12475 C0SZ6Q 44347005 Ki = 57 nM T12475 CMZ67A 44347047 Ki = 8 nM T12475 CN5P7O 44347048 Ki = 56 nM T12475 C2UAY6 44347085 Ki = 10 nM T12475 CQHO57 44352512 IC50 = 0.4 nM T12475 CRD59K 44352513 Ki = 2100 nM T12475 CN2WM6 44352514 Ki = 2500 nM T12475 CK28SX 44352515 Ki = 260 nM T12475 C5CJP7 44352548 Ki = 2400 nM T12475 C3KT4B 44352566 Ki = 28000 nM T12475 CBLM03 44352573 Ki > 50000 nM T12475 C2QG7F 44352607 Ki = 400 nM T12475 C7Y3LI 44352608 Ki > 50000 nM T12475 CI16VP 44352609 Ki > 50000 nM T12475 C5F7XC 44352641 Ki = 6600 nM T12475 CKN0W6 44352652 Ki = 31 nM T12475 CM4GZ2 44352657 Ki = 33 nM T12475 C7ATX0 44352665 Ki = 180 nM T12475 CNG67A 44352678 Ki = 400 nM T12475 CQFR35 44352679 Ki = 800 nM T12475 C60YZR 44352734 Ki = 1200 nM T12475 CQC83V 44352735 Ki = 2200 nM T12475 CZ7MX1 44352747 Ki = 42000 nM T12475 CA12CZ 44352801 Ki = 2000 nM T12475 CM26XR 44352874 Ki = 2600 nM T12475 CBI1T2 44352933 Ki = 3700 nM T12475 C1P0SI 44352942 Ki = 8500 nM T12475 CC9U8D 44352949 Ki = 6000 nM T12475 CCF53D 44352957 Ki = 4900 nM T12475 C1T8HR 44352975 Ki > 50000 nM T12475 C0ZQ4F 44353200 Ki = 32 nM T12475 C7XF6D 44353201 Ki = 10 nM T12475 CMCG71 44353228 Ki = 4 nM T12475 CY29JH 44353229 Ki = 100 nM T12475 C65JBG 44353230 Ki = 14 nM T12475 CW5V8T 44353231 Ki = 62 nM T12475 CGKR09 44353238 Ki = 400 nM T12475 CBKV32 44353246 Ki = 190 nM T12475 C5EM0B 44353247 Ki = 44 nM T12475 C8K5QV 44353248 Ki = 1.2 nM T12475 C5T7QJ 44353249 Ki = 5.8 nM T12475 CH7U2X 44353254 Ki = 130 nM T12475 C3Q7UD 44353258 Ki = 3.8 nM T12475 C83BTF 44353262 Ki = 2.1 nM T12475 C2NZQ3 44353263 Ki = 64 nM T12475 CXAD84 44353264 Ki = 270 nM T12475 CK95NX 44353265 Ki = 440 nM T12475 CO68AE 44353266 Ki = 154 nM T12475 CJ6E0H 44353270 Ki = 14 nM T12475 CI92CJ 44353271 Ki = 42 nM T12475 CE1L4R 44353276 Ki = 17 nM T12475 CF4DJ0 44353277 Ki = 1.1 nM T12475 CZ37PB 44353284 Ki = 630 nM T12475 C81UZX 44353285 Ki = 3.3 nM T12475 C0OR7I 44353288 Ki = 9.2 nM T12475 CB0G7U 44353304 Ki = 21 nM T12475 CK47NB 44353305 Ki = 450 nM T12475 CRT73O 44361351 IC50 = 7.9 nM T12475 CD8B7P 44361468 IC50 = 7.7 nM T12475 C7XSN2 44361524 IC50 = 13 nM T12475 C3ILW4 44361587 IC50 = 8.8 nM T12475 C2AV6H 44361795 IC50 = 2.8 nM T12475 C91MSF 44361796 IC50 = 5.8 nM T12475 C37RVW 44361797 IC50 = 7.9 nM T12475 CA78JT 44361802 IC50 = 6.4 nM T12475 CRQ6N8 44361888 IC50 = 10.8 nM T12475 CJ31OK 44379747 Ki = 14 nM T12475 C4X3SP 44380146 IC50 = 1.1 nM T12475 C0C1LJ 44380147 IC50 = 5 nM T12475 C8ZG2P 44380148 IC50 = 3.6 nM T12475 C5H6TG 44380192 IC50 = 15.3 nM T12475 C0YSC9 44380212 IC50 = 2.4 nM T12475 C61CGF 44380222 IC50 = 0.8 nM T12475 CY1RF0 44380236 IC50 = 0.6 nM T12475 C9C5FR 44380317 IC50 = 2.1 nM T12475 CTDC79 44380318 IC50 = 1.1 nM T12475 CZ5TK1 44380319 IC50 = 46.4 nM T12475 CQ05NO 44380394 IC50 = 0.4 nM T12475 C8BO2Z 44380466 Ki = 0.14 nM T12475 C3R9FW 44380478 IC50 = 0.7 nM T12475 C7U1XT 44380483 IC50 = 0.7 nM T12475 CUR9A5 44380487 IC50 = 1.5 nM T12475 CKY1Q3 44380488 IC50 = 0.3 nM T12475 C6INE9 44380512 IC50 = 0.6 nM T12475 C31ZHW 44380513 IC50 = 0.7 nM T12475 C15CFE 44380514 IC50 = 0.4 nM T12475 CC0EA3 44380536 IC50 = 0.6 nM T12475 C8J6QW 44380537 IC50 = 0.4 nM T12475 C4T3JB 44380538 IC50 = 0.5 nM T12475 CS7BV5 44380551 IC50 = 3 nM T12475 CD76UJ 44380552 IC50 = 2.1 nM T12475 C94JQT 44380624 IC50 = 16.5 nM T12475 C16VXA 44380625 IC50 = 0.3 nM T12475 C4FT3G 44380626 IC50 = 0.4 nM T12475 CW4M9S 44380643 IC50 = 0.3 nM T12475 CDAE02 44380658 Ki = 0.32 nM T12475 C7DA2K 44380681 IC50 = 0.9 nM T12475 CU2EP8 44380796 IC50 = 0.6 nM T12475 CJN6K7 44380797 IC50 = 1.5 nM T12475 CK4A6Q 44380798 IC50 = 0.6 nM T12475 C8NB1T 44387880 Ki = 120 nM T12475 CV1O8G 44387883 Ki = 620 nM T12475 C64JEC 44387885 Ki = 1500 nM T12475 CM0P8L 44387888 Ki = 66 nM T12475 CVO24X 44387891 Ki > 10000 nM T12475 C4GBW2 44387896 Ki = 9 nM T12475 C5HNA6 44387898 Ki = 75 nM T12475 CLHA03 44387907 Ki = 20 nM T12475 CGKY89 44387908 Ki = 27 nM T12475 CS1LK9 44387909 Ki = 580 nM T12475 CT47HC 44387918 Ki = 29 nM T12475 CJB4X8 44387920 Ki = 800 nM T12475 C67VEO 44387922 Ki = 83 nM T12475 CW3OZ5 44387924 Ki = 11 nM T12475 CJ9ZS6 44387926 Ki = 180 nM T12475 COZ12K 44387935 Ki = 28 nM T12475 CB2Y6T 44387945 Ki = 70 nM T12475 C9P5TC 44387961 Ki = 18 nM T12475 CKU05A 44387972 Ki = 5 nM T12475 CJ1V8X 44387977 Ki = 3 nM T12475 CYP7N1 44387979 Ki = 120 nM T12475 C6IT7U 44387988 Ki = 36 nM T12475 C9IC3Q 44387992 Ki = 20 nM T12475 CE23JP 44388002 Ki = 24 nM T12475 CG60VU 44388009 Ki = 630 nM T12475 CHQ2G9 44388018 Ki = 13 nM T12475 C6SAE2 44388026 Ki = 73 nM T12475 CR9O0C 44388033 Ki = 66 nM T12475 CDGT03 44388510 Ki = 0.5 nM T12475 C3X1UK 44388511 Ki = 3.9 nM T12475 C3U9VL 44389571 Ki = 460 nM T12475 CX78WH 44389647 Ki = 870 nM T12475 C3X7HL 44389652 Ki = 125 nM T12475 CB4KC8 44389658 Ki = 110 nM T12475 C08VHB 44390758 Ki = 89 nM T12475 C7AXB1 44390769 Ki = 220 nM T12475 CR9XQ4 44390780 Ki = 410 nM T12475 CCK4F2 44390795 Ki = 380 nM T12475 CIS49X 44390818 Ki > 20000 nM T12475 CTE6F4 44391498 IC50 = 5800 nM T12475 CFEP75 44391499 IC50 = 300 nM T12475 COT84R 44391510 IC50 = 4800 nM T12475 C4R6BS 44391511 IC50 > 10000 nM T12475 CLF4Y8 44391516 IC50 = 220 nM T12475 CZ98WM 44391525 IC50 = 1100 nM T12475 CR86IW 44391526 IC50 = 670 nM T12475 C76TAB 44391541 IC50 = 1100 nM T12475 C59JAO 44391542 IC50 = 820 nM T12475 C0C7IO 44391548 IC50 = 280 nM T12475 CPLJ78 44391554 IC50 > 10000 nM T12475 CXT48Y 44391566 IC50 = 250 nM T12475 C5JRI2 44391574 IC50 = 1400 nM T12475 CH41FJ 44391612 IC50 = 270 nM T12475 C8O2PH 44391613 IC50 = 2100 nM T12475 CR4I8Z 44391628 IC50 = 490 nM T12475 CSU23B 44391653 IC50 > 10000 nM T12475 CGL16J 44391670 IC50 = 880 nM T12475 CMW8K0 44391692 IC50 = 390 nM T12475 CPHX28 44391693 IC50 = 57 nM T12475 C9DZN1 44391703 IC50 = 66 nM T12475 CL52EN 44391714 IC50 = 320 nM T12475 C2O3UD 44391718 IC50 = 150 nM T12475 CZ3H4T 44391728 IC50 = 230 nM T12475 CHY9S7 44391734 IC50 = 690 nM T12475 C9UD8M 44391735 IC50 = 83 nM T12475 C7S9DN 44391752 IC50 = 20 nM T12475 C5PQR7 44391754 IC50 = 490 nM T12475 C3PA7C 44391767 IC50 > 10000 nM T12475 C2V5YU 44391771 IC50 = 180 nM T12475 C2XH5W 44391784 IC50 = 400 nM T12475 C8UY5V 44391807 IC50 > 10000 nM T12475 CXOZ68 44391808 IC50 = 22 nM T12475 CTM2S4 44391821 IC50 = 740 nM T12475 C0IW4A 44391826 IC50 = 340 nM T12475 C3FNB1 44391835 IC50 = 2600 nM T12475 C78NTV 44391849 IC50 = 1900 nM T12475 C5E4IX 44394567 Ki = 14 nM T12475 C43NCH 44394577 Ki = 210 nM T12475 C4TEK2 44394578 Ki = 500 nM T12475 C5W8FE 44394589 Ki = 10 nM T12475 CLH7X0 44394608 Ki = 49 nM T12475 CVZ39D 44394614 Ki = 35 nM T12475 CDP67J 44394615 Ki = 20 nM T12475 C35POC 44394616 Ki = 7 nM T12475 CMO24B 44394649 Ki = 34 nM T12475 CST3R9 44394651 Ki = 130 nM T12475 CZM2J0 44394661 Ki = 15 nM T12475 CJR6I8 44394685 Ki = 130 nM T12475 C6ZOD2 44394714 Ki = 160 nM T12475 CAVG82 44394723 Ki = 120 nM T12475 C6OPK5 44394753 Ki = 150 nM T12475 CKS6B0 44394767 Ki = 42 nM T12475 C5ISK4 44394768 Ki = 33 nM T12475 C85YDH 44394778 Ki = 9 nM T12475 CI5F2O 44394779 Ki = 47 nM T12475 CN35MY 44394818 Ki = 26 nM T12475 C7N2ZE 44394835 Ki = 1500 nM T12475 CH9A1L 44394841 Ki = 49 nM T12475 C95TAB 44394852 Ki = 270 nM T12475 C1KHJ8 44394857 Ki = 18 nM T12475 CF31WT 44394893 Ki = 3000 nM T12475 C7TVS1 44394894 Ki = 42 nM T12475 CK3SE0 44394896 Ki = 70 nM T12475 CE32VZ 44394901 Ki = 30 nM T12475 CG7ZT8 44395435 IC50 = 0.32 nM T12475 C49RQL 44395462 IC50 = 0.55 nM T12475 CJ15UQ 44395463 IC50 = 2 nM T12475 CALH48 44395491 IC50 = 0.8 nM T12475 CB05VD 44395502 IC50 = 0.7 nM T12475 CT1F3L 44395533 IC50 = 0.6 nM T12475 CK2F3E 44395583 IC50 = 49 nM T12475 CGZ9V2 44395623 IC50 = 0.3 nM T12475 C3O1QY 44395650 IC50 = 1.3 nM T12475 CAB59T 44395677 IC50 = 1.4 nM T12475 CP6GJ9 44398001 IC50 = 1.98 nM T12475 C73OZF 44398040 IC50 = 2.85 nM T12475 CB6U3S 44398043 IC50 = 1.62 nM T12475 CRW98K 44398044 IC50 = 2.24 nM T12475 C8OT4L 44398045 IC50 = 1.77 nM T12475 CO9S5F 44398046 IC50 = 1.85 nM T12475 CUBJ08 44398047 IC50 = 1.47 nM T12475 C7W0UO 44398063 IC50 = 1.56 nM T12475 C3L4HN 44398064 IC50 = 1.54 nM T12475 C2TVL4 44398065 IC50 = 1.5 nM T12475 CP4W2T 44398066 IC50 = 1.77 nM T12475 CVN17W 44398086 IC50 = 52.24 nM T12475 C92VFH 44398117 IC50 = 13.47 nM T12475 CBK69Y 44398118 IC50 = 9.18 nM T12475 CIE64L 44398119 IC50 = 25.79 nM T12475 CIY7Q5 44398120 IC50 = 48.91 nM T12475 CBEO08 44398135 IC50 = 1.97 nM T12475 C5TWQ9 44398149 IC50 = 178.19 nM T12475 CJ5RS1 44398150 IC50 = 1.72 nM T12475 CHA01F 44398151 IC50 = 1.83 nM T12475 CBZ98L 44398152 IC50 = 1.38 nM T12475 CH3V4J 44398178 IC50 = 2.71 nM T12475 CJ3MI9 44398179 IC50 = 3.79 nM T12475 CMA94R 44398180 IC50 = 4.25 nM T12475 CH27CV 44398181 IC50 = 5.52 nM T12475 C3QOA9 44398182 IC50 = 3.5 nM T12475 C0WVI8 44398395 IC50 = 5.31 nM T12475 CP2N9S 44398396 IC50 = 22.58 nM T12475 CN91AI 44399944 Ki = 5.3 nM T12475 C2R9ZB 44399956 Ki = 570 nM T12475 C6CPF7 44400099 Ki = 19 nM T12475 C50MUR 44400121 Ki = 7.8 nM T12475 CCZS53 44400122 Ki = 660 nM T12475 C28TXH 44400146 Ki = 120 nM T12475 C1LMC3 44400147 Ki = 1400 nM T12475 C0ST3Y 44400187 Ki = 4 nM T12475 CDZ7C9 44400188 Ki = 8 nM T12475 CKJ0R4 44400195 Ki = 55 nM T12475 CXMZ97 44400204 Ki = 18 nM T12475 C6C5FX 44400229 Ki = 1.4 nM T12475 C5YS3K 44400230 Ki = 6 nM T12475 CLIK31 44400235 Ki = 0.6 nM T12475 COVG03 44400245 Ki = 0.9 nM T12475 C7J3YU 44400246 Ki = 30 nM T12475 CB5W2F 44400247 Ki = 9.1 nM T12475 CDA2G8 44400255 Ki = 3100 nM T12475 C68TAQ 44400261 Ki = 1.3 nM T12475 CL7A1W 44400271 Ki = 1 nM T12475 C59YMH 44400350 Ki = 2.6 nM T12475 CL85GS 44400352 Ki = 1.8 nM T12475 CDC8P7 44400353 Ki = 8.2 nM T12475 C98DUH 44400354 Ki = 6.3 nM T12475 C8XE3Z 44402038 IC50 = 880 nM T12475 C87LQO 44402057 IC50 = 57 nM T12475 CV38UX 44402072 IC50 = 250 nM T12475 CS64QR 44402105 IC50 = 360 nM T12475 C1ZI0P 44402232 IC50 = 1500 nM T12475 C6A3ZW 44402256 IC50 = 28 nM T12475 CG5EA9 44402273 IC50 = 180 nM T12475 CNG9K1 44402293 IC50 = 43 nM T12475 C7J1DT 44402335 IC50 = 180 nM T12475 C0QX7G 44402360 IC50 = 350 nM T12475 C9PV2W 44402377 IC50 = 6500 nM T12475 CA21YV 44402378 IC50 = 600 nM T12475 CJ7L8H 44402395 IC50 = 2.37 nM T12475 CQT0S6 44402396 IC50 = 6.31 nM T12475 CL8VO0 44402397 IC50 = 6.31 nM T12475 C5D0VR 44402398 IC50 = 2.82 nM T12475 C8V7KC 44402403 IC50 = 21 nM T12475 C0K4FZ 44402404 IC50 = 610 nM T12475 CW59LA 44402405 IC50 = 2100 nM T12475 C47PUC 44402426 IC50 = 1900 nM T12475 C02WKU 44402431 IC50 = 280 nM T12475 CA18SB 44402462 IC50 = 6300 nM T12475 CBWC25 44402463 IC50 = 42 nM T12475 CL1W8N 44402464 IC50 = 61 nM T12475 CYA4E3 44402465 IC50 = 69 nM T12475 C0TC3F 44402466 IC50 = 31 nM T12475 CO29PL 44402467 IC50 = 130 nM T12475 CPZU59 44402468 IC50 = 160 nM T12475 CV8U3B 44402469 IC50 = 170 nM T12475 CR30VC 44402470 IC50 = 260 nM T12475 CT2SL0 44402471 IC50 = 23 nM T12475 CFB54Y 44402472 IC50 = 27 nM T12475 CM85ZQ 44402492 IC50 = 33 nM T12475 CB9T3S 44402499 IC50 = 47 nM T12475 CIP9E4 44402518 IC50 = 1.995 nM T12475 C3VNE6 44402538 IC50 = 62 nM T12475 CK0A7Q 44402553 IC50 = 37 nM T12475 C2B1GK 44402560 IC50 = 160 nM T12475 CI46SK 44402571 IC50 = 3200 nM T12475 C2NI6G 44402572 IC50 = 3300 nM T12475 CJ2V0R 44402589 IC50 = 270 nM T12475 C89HOR 44402616 IC50 = 79 nM T12475 C3OF2P 44402638 IC50 = 3.162 nM T12475 C4YZ1N 44402639 IC50 = 1.85 nM T12475 C3GY0J 44402640 IC50 = 1.78 nM T12475 CS6LU1 44402645 IC50 = 41 nM T12475 C3XQD0 44402646 IC50 = 410 nM T12475 C9KQ0F 44402647 IC50 = 120 nM T12475 C50FVK 44402648 IC50 = 980 nM T12475 C05KJS 44402649 IC50 = 190 nM T12475 CR15JA 44402670 IC50 = 210 nM T12475 CEGT74 44402672 IC50 = 570 nM T12475 C2SWC1 44402673 IC50 = 210 nM T12475 CY9K5I 44402759 IC50 = 2.46 nM T12475 CGD16R 44406776 IC50 = 3.7 nM T12475 CNR6O3 44411993 IC50 = 0.7 nM T12475 CCN94V 44412054 IC50 = 1.514 nM T12475 C7TCZ3 44412876 IC50 = 700 nM T12475 C6LJE5 44412890 IC50 = 0.6 nM T12475 CAV19O 44412945 IC50 = 1 nM T12475 CK8H9N 44412946 IC50 = 30 nM T12475 C08FVY 44412947 IC50 = 2 nM T12475 CW62ND 44412978 IC50 = 500 nM T12475 C1T2BH 44413009 IC50 = 40 nM T12475 CTZS42 44413029 IC50 = 10 nM T12475 CT6B5Z 44413066 IC50 = 2 nM T12475 C4S7TI 44413067 IC50 = 0.4 nM T12475 CH5QT9 44417614 IC50 = 70 nM T12475 CT4QR9 44417615 IC50 = 800 nM T12475 C0F3MG 44432626 IC50 > 10000 nM T12475 CX6Q1V 44432627 IC50 = 8090 nM T12475 CH1UD0 44432628 IC50 = 3480 nM T12475 CS50LE 44432635 IC50 = 475 nM T12475 CFV79O 44432636 IC50 = 546 nM T12475 C4SCA7 44432637 IC50 > 10000 nM T12475 CPTV07 44432638 IC50 = 1110 nM T12475 CGF71S 44432639 IC50 = 462 nM T12475 C3YWK5 44432640 IC50 = 271 nM T12475 C3S9RA 44432641 IC50 = 267 nM T12475 CQ46LO 44432642 IC50 = 86 nM T12475 CNQ3R8 44432643 IC50 = 62 nM T12475 CXCK53 44432645 IC50 = 4180 nM T12475 C7T1NP 44432646 IC50 = 205 nM T12475 CPM79H 44432647 IC50 = 32 nM T12475 CWZL59 44432648 IC50 = 60 nM T12475 CCQG31 44432649 IC50 = 87 nM T12475 CQT3Z0 44432650 IC50 = 91 nM T12475 CB8R9X 44432651 IC50 = 26 nM T12475 CS6WI8 44432652 IC50 = 9 nM T12475 C5M0UD 44432653 IC50 = 16 nM T12475 CB3R7Y 44432654 IC50 = 7 nM T12475 CZLJ29 44432655 IC50 = 63 nM T12475 CU5GE9 44432656 IC50 = 1600 nM T12475 CPS64W 44432657 IC50 = 22 nM T12475 CNDE50 44433200 Ki = 540 nM T12475 C0B2HJ 44434373 Ki = 162.18 nM T12475 CI1U8W 44434374 IC50 < 10000 nM T12475 CE0AD7 44434375 IC50 < 10000 nM T12475 C9W1MK 44434376 IC50 < 10000 nM T12475 C4VL3D 44434377 IC50 < 10000 nM T12475 CXEI96 44434378 IC50 < 10000 nM T12475 CHXQ70 44434381 IC50 < 10000 nM T12475 CS6OH2 44434382 IC50 < 10000 nM T12475 C5P3ZC 44434383 IC50 < 10000 nM T12475 C1NS9Z 44434384 IC50 < 10000 nM T12475 CH62LS 44434385 IC50 < 10000 nM T12475 C68XDJ 44434386 Ki = 1.349 nM T12475 CQL64Z 44434387 IC50 = 2570.4 nM T12475 CAUS34 44434388 IC50 = 3630.78 nM T12475 C92GBQ 44434389 IC50 = 2398.83 nM T12475 CPRH80 44434390 IC50 = 3019.95 nM T12475 CLU28X 44434391 IC50 = 676.08 nM T12475 CN07XM 44434392 IC50 = 1905.46 nM T12475 CBLU65 44434402 IC50 = 3162.28 nM T12475 C3BCG9 44434404 Ki = 23.44 nM T12475 CV1TD4 44434411 Ki = 29.51 nM T12475 C4PJW7 44434412 IC50 = 1348.96 nM T12475 C1NSZ0 44434414 Ki = 5.248 nM T12475 C31RJW 44434415 IC50 = 724.44 nM T12475 C89LIS 44434428 IC50 = 524.81 nM T12475 CA49FW 44434431 IC50 = 467.74 nM T12475 C5BIX8 44434432 IC50 = 724.44 nM T12475 COC13L 44434433 IC50 = 831.76 nM T12475 C5W6JY 44434434 IC50 = 1905.46 nM T12475 C31TQH 44434435 IC50 = 1548.82 nM T12475 CM7P4I 44434436 Ki = 58.88 nM T12475 C9JD3V 44434437 Ki = 69.18 nM T12475 CS10BH 44434438 Ki = 194.98 nM T12475 CD4Q3W 44435817 Ki = 1290 nM T12475 COJ7Z3 44435818 Ki = 970 nM T12475 CAL2P0 44435819 Ki = 1580 nM T12475 CN8D3W 44435820 Ki = 2200 nM T12475 CBE01S 44435821 Ki > 10000 nM T12475 CEBU80 44435822 Ki = 980 nM T12475 CO5WV4 44435825 Ki = 990 nM T12475 C7EJ5N 44435826 Ki > 10000 nM T12475 CE8G4O 44435827 Ki > 10000 nM T12475 CN6D2K 44435828 Ki = 515 nM T12475 C6GOU4 44435829 Ki = 35 nM T12475 CR04XY 44435973 Ki > 10000 nM T12475 C2AP1R 44435975 Ki = 20 nM T12475 C1IM6U 44435976 Ki = 300 nM T12475 C9ZGE6 44435977 Ki = 17 nM T12475 CEP45X 44435978 Ki = 100 nM T12475 CTDJ76 44435979 Ki = 10 nM T12475 CD9WG1 44435980 Ki = 30 nM T12475 CM64FI 44435981 Ki = 805 nM T12475 CGZC73 44435982 Ki = 15 nM T12475 CW4A0H 44435983 Ki = 850 nM T12475 C9YJ4E 44435984 Ki = 85 nM T12475 CY8MS9 44435985 Ki = 255 nM T12475 CR1O7E 44435986 Ki = 15 nM T12475 CL8Q9M 44435987 Ki > 10000 nM T12475 CU47OL 44435988 Ki > 10000 nM T12475 CE2QH3 44435989 Ki > 10000 nM T12475 C8FH9K 44435990 Ki = 380 nM T12475 C2C1IQ 44435991 Ki = 305 nM T12475 CH46ZR 44435992 Ki = 80 nM T12475 C97RFB 44435993 Ki = 10 nM T12475 CSYH19 44435994 Ki = 1400 nM T12475 C54OPY 44435995 Ki = 1800 nM T12475 CISP05 44435996 Ki = 180 nM T12475 CIT03Z 44435997 Ki > 10000 nM T12475 CNW62E 44435998 Ki = 1710 nM T12475 C1MKW2 44435999 Ki = 2590 nM T12475 CT2DX9 44436000 Ki = 520 nM T12475 CH7O9L 44436001 Ki = 945 nM T12475 C2Q5YM 44436002 Ki = 25 nM T12475 CS8I5A 44436003 Ki = 30 nM T12475 CX1D6V 44436004 Ki = 2410 nM T12475 CGR72I 44436005 Ki = 2450 nM T12475 C2CQV7 44436006 Ki > 10000 nM T12475 C6KV0L 44436007 Ki > 10000 nM T12475 CGC24A 44436008 Ki = 2580 nM T12475 CK7Q8Y 44436009 Ki = 160 nM T12475 CV94OL 44436010 Ki = 490 nM T12475 CF8V4P 44436011 Ki = 600 nM T12475 CW8RE9 44436013 Ki > 10000 nM T12475 CS14DQ 44436014 Ki = 1370 nM T12475 CZ98VY 44436015 Ki = 20 nM T12475 C9Y3EZ 44436016 Ki = 1370 nM T12475 CV9NT3 44436017 Ki = 10 nM T12475 CH20CE 44436018 Ki = 45 nM T12475 CY3Z7T 44436019 Ki = 70 nM T12475 CVD86R 44444617 IC50 = 244 nM T12475 C0UR9E 44444626 IC50 = 3 nM T12475 C3X1DG 44444628 IC50 = 12 nM T12475 CTX79C 44444630 IC50 = 96 nM T12475 CO8KR1 44444632 IC50 = 2 nM T12475 CASL32 44444635 IC50 = 56 nM T12475 CH6E1P 44444639 IC50 = 209 nM T12475 C9GIR7 44444641 IC50 = 161 nM T12475 C3MG0L 44444642 IC50 = 197 nM T12475 C3BX9Y 44444644 IC50 = 696 nM T12475 CAMH23 44444645 IC50 = 345 nM T12475 CVRZ54 44444647 IC50 = 280 nM T12475 CBZ9S3 44444649 IC50 = 171 nM T12475 C8V0SW 44444652 IC50 = 178 nM T12475 C79TVN 44444663 IC50 = 743 nM T12475 CPQW62 44444665 IC50 = 111 nM T12475 CU58SE 44444668 IC50 = 238 nM T12475 C6L3KV 44444670 IC50 = 214 nM T12475 CU3V2K 44444672 IC50 = 173 nM T12475 C0JC2Y 44444673 IC50 = 184 nM T12475 CPI6R7 44444675 IC50 = 88 nM T12475 C0G9FY 44444676 IC50 = 117 nM T12475 C1AF7Z 44444678 IC50 = 33 nM T12475 CWXR27 44448860 Ki = 68 nM T12475 C5D1WQ 44448991 Ki = 0.7 nM T12475 CO2XN4 44449095 Ki = 3.7 nM T12475 CXLN43 44449120 Ki = 0.3 nM T12475 CLY90R 44449153 Ki = 7.4 nM T12475 C4B9ZH 44449156 Ki = 4.2 nM T12475 CG9BY0 44449186 Ki = 20 nM T12475 CF81TQ 44449681 Ki = 0.61 nM T12475 CNM1X9 44449682 Ki = 4.5 nM T12475 CMO4U0 44449683 Ki = 4.9 nM T12475 CQ7PC6 44451258 Ki = 850 nM T12475 C83VTS 44451276 Ki = 480 nM T12475 CA36SN 44451294 Ki = 700 nM T12475 CORX87 44451319 Ki = 260 nM T12475 CDY86U 44451331 Ki = 3200 nM T12475 C3NI0S 44451342 Ki = 380 nM T12475 CYC3J1 44451343 Ki = 840 nM T12475 C09WDB 44451345 Ki = 530 nM T12475 C8UA2K 44451349 Ki = 1900 nM T12475 C94CLQ 44451350 Ki = 50 nM T12475 C23MDG 44451355 Ki = 0.7 nM T12475 COL9E6 44451356 Ki = 580 nM T12475 CZM37I 44451367 Ki = 110 nM T12475 CVQ3I0 44451379 IC50 = 520 nM T12475 CI15FA 44451385 Ki = 2500 nM T12475 CL27UG 44451391 Ki = 510 nM T12475 CN5EO1 44451396 Ki = 170 nM T12475 CF6O2B 44451397 IC50 = 1100 nM T12475 CB5Q0H 44451398 Ki = 3300 nM T12475 CE5ZB6 44451399 Ki = 400 nM T12475 CIPJ67 44451406 Ki = 4400 nM T12475 C4T1IZ 44451408 Ki = 740 nM T12475 CO9P2W 44451418 Ki = 3000 nM T12475 C7YDZ5 44451419 Ki = 930 nM T12475 CZ5Y0V 44451420 Ki = 620 nM T12475 CCV0E2 44451430 Ki = 930 nM T12475 CQI3G0 44451446 Ki = 820 nM T12475 CT51RZ 44451447 Ki = 600 nM T12475 CTZO29 44451460 Ki = 2200 nM T12475 C5PS3J 44451474 Ki = 5300 nM T12475 C2K7IV 44451476 Ki = 1000 nM T12475 CVF08D 44451485 Ki = 1100 nM T12475 CN91FU 44451486 Ki = 720 nM T12475 C75SYB 44451498 Ki = 500 nM T12475 CCYP84 44460342 IC50 = 0.5 nM T12475 CZ2CI5 44460343 IC50 = 0.7 nM T12475 CB23PH 44560995 IC50 = 1500 nM T12475 C0N1LV 44561105 IC50 = 3300 nM T12475 CM8IS1 44561108 IC50 = 9500 nM T12475 CWT1X2 44561141 IC50 = 3400 nM T12475 C4SW8J 44561142 IC50 = 4500 nM T12475 CV78LP 44561265 IC50 = 6300 nM T12475 C9BLD8 44561368 IC50 = 8.7 nM T12475 CE1V2F 44561369 IC50 = 5.7 nM T12475 C1TFD7 44561397 IC50 = 5.5 nM T12475 C9ARN8 44572235 IC50 = 3.5 nM T12475 C0CPE6 44572236 IC50 = 14 nM T12475 CNA0Z9 44572286 IC50 = 16 nM T12475 CN9MT5 44572287 IC50 = 24 nM T12475 CQE6V2 44573110 IC50 = 10 nM T12475 CZ0Y5K 44573111 IC50 = 18 nM T12475 C5GH0O 44573112 IC50 = 26 nM T12475 CMXJ54 44573113 IC50 = 10 nM T12475 CXW23Z 44573275 IC50 = 11 nM T12475 C9BC7A 44573276 IC50 = 8 nM T12475 C1TDC2 44573277 IC50 = 29 nM T12475 C7Q0SA 44573278 IC50 = 57 nM T12475 C1B0KY 44573507 IC50 = 705 nM T12475 CE3DV9 44573585 IC50 = 90 nM T12475 CE6KZ9 44573586 IC50 = 31 nM T12475 C3S1FB 44573625 IC50 = 37 nM T12475 CSG8P3 44573626 IC50 = 27 nM T12475 CDQ4Y6 44573627 IC50 = 27 nM T12475 CKW2P1 44573628 IC50 = 20 nM T12475 CUH2K6 44573670 IC50 = 21 nM T12475 C2R6HW 44573713 IC50 = 23 nM T12475 C06TLX 44573714 IC50 = 68 nM T12475 C12QRZ 44573753 IC50 = 83 nM T12475 CM2Z6Y 44573789 IC50 = 12 nM T12475 CH5M3I 44573790 IC50 = 19 nM T12475 C3A2EJ 44573791 IC50 = 71 nM T12475 CTA0G9 44576642 Ki = 69 nM T12475 CLE52Y 44576643 Ki = 1100 nM T12475 CV4HU0 44576644 Ki = 3.3 nM T12475 C74QBS 44576645 Ki = 10 nM T12475 CVZ2A9 44576655 Ki = 77 nM T12475 C32ANR 44576656 IC50 = 7900 nM T12475 C38AKC 44576657 Ki = 3700 nM T12475 C9IB4V 44576677 Ki > 10000 nM T12475 CY1KQ8 44576678 Ki = 66 nM T12475 CRS2A0 44576679 Ki = 22 nM T12475 CMZ6C1 44576680 Ki = 3.4 nM T12475 CSIH37 44576681 Ki = 42 nM T12475 C48CGJ 44577051 Ki = 23 nM T12475 CAFQ96 44577067 Ki = 220 nM T12475 C5AL2O 44577069 IC50 = 3400 nM T12475 CSX73A 44577096 Ki = 34 nM T12475 C5HC7Z 44577097 Ki = 14 nM T12475 CO7W1K 44577098 Ki = 4.4 nM T12475 CLG0Q1 44577099 Ki = 40 nM T12475 CAZ7U0 44577100 Ki = 580 nM T12475 C2HT3J 44577101 Ki = 13 nM T12475 C0WS7X 44577102 IC50 = 10000 nM T12475 C01TVM 44577103 IC50 = 41000 nM T12475 C78YXI 44577104 IC50 = 6.6 nM T12475 CY2WG3 44587391 Ki = 34 nM T12475 CZ35WG 44587392 Ki = 33 nM T12475 CDIQ98 44587393 Ki = 4.1 nM T12475 C81XUZ 44587394 Ki = 7.5 nM T12475 CP8EC7 44587395 Ki = 4.7 nM T12475 CP5S0E 44587396 Ki = 10.1 nM T12475 CK47QS 44587397 Ki = 52 nM T12475 C72XPL 44587398 Ki = 15 nM T12475 CO96FR 44587399 Ki = 27 nM T12475 CCU14T 44587400 Ki = 98 nM T12475 CAO71W 44587401 Ki = 155 nM T12475 C5O1CZ 44587402 Ki = 35 nM T12475 CA7FG6 44587403 Ki = 9.3 nM T12475 C37JHB 44587404 Ki = 38 nM T12475 CSZ7D4 44587405 Ki = 29 nM T12475 CR8T7B 44593415 IC50 = 790 nM T12475 C0RQH9 44593424 IC50 = 9.4 nM T12475 CY75PU 44593425 IC50 = 4 nM T12475 CEFN61 44593613 Ki = 110 nM T12475 CQ3U9E 44593614 Ki = 3900 nM T12475 CIMG71 44593615 Ki = 32 nM T12475 CL2T6A 49796662 IC50 = 130 nM T12475 CK69HN 49796663 IC50 = 40 nM T12475 CL5R4J 49796664 IC50 = 7 nM T12475 C21QVT 49796665 IC50 = 3.8 nM T12475 C4BL5D 49796666 IC50 = 110 nM T12475 CMAD14 49796667 IC50 = 190 nM T12475 CM5I0J 49796668 IC50 = 45 nM T12475 C89WLS 49796669 IC50 = 15 nM T12475 CQ1D3M 49796670 IC50 = 9 nM T12475 CBA6W2 49796671 IC50 = 1.8 nM T12475 C28TMR 49796672 IC50 = 1.4 nM T12475 C0U1JE 49796673 IC50 = 2.3 nM T12475 CY6W7R 49796674 IC50 = 860 nM T12475 C9F3UH 49796675 IC50 = 22 nM T12475 CI3Q9O 49796676 IC50 = 320 nM T12475 C26SNP 49796677 IC50 = 290 nM T12475 COPT75 49796678 IC50 = 28 nM T12475 CLT32V 49796679 IC50 = 3.6 nM T12475 CQ84ZY 49796680 IC50 = 23 nM T12475 CJ5OD1 49796681 IC50 = 10.9 nM T12475 CD1M9A 49796682 IC50 = 2.8 nM T12475 CFP31J 49796683 IC50 = 2.9 nM T12475 CW2JM9 53238728 IC50 = 12 nM T12475 CSL7D0 53238731 IC50 = 14 nM T12475 C2FE7P 53238732 IC50 > 100 nM T12475 CBFM18 53239181 IC50 = 10 nM T12475 C14FZD 53239183 IC50 = 8.96 nM T12475 CU64VQ 53239184 IC50 = 48 nM T12475 C61WUG 53239400 IC50 > 300 nM T12475 CL2G4N 53239401 IC50 > 300 nM T12475 CW0YI7 53239615 IC50 = 2.76 nM T12475 CEP1K5 53239616 IC50 > 300 nM T12475 CHOE79 53386756 IC50 = 0.2 nM T12475 C9CWM3 53386757 IC50 = 0.37 nM T12475 CL4O7B 53386758 IC50 = 0.3 nM T12475 C5CJH6 53386914 IC50 = 0.3 nM T12475 CKBL02 53386915 IC50 = 0.1 nM T12475 C3VI7B 53386916 IC50 = 1 nM T12475 C2OL0W 53386917 IC50 = 0.2 nM T12475 C61ZLR 53387071 IC50 = 0.24 nM T12475 C76XAU 53388958 IC50 = 0.08 nM T12475 CLM14F 53388959 IC50 = 0.2 nM T12475 CP8G1I 53388960 IC50 = 0.07 nM T12475 C1EPL3 53389115 IC50 = 0.24 nM T12475 C9TN5J 53389116 IC50 = 0.3 nM T12475 C8DZV1 53389117 IC50 = 0.09 nM T12475 CYTI51 53389118 IC50 = 0.2 nM T12475 CWM12T 54582417 IC50 = 3.2 nM T12475 CF3ED5 54584354 IC50 = 2440 nM T12475 C9JE4A 56655880 IC50 = 22.87 nM T12475 CR9CJ6 58239302 IC50 = 0.58 nM T12475 C0YU9A 67142711 IC50 = 19.1 nM T12475 C12VTJ 67142732 IC50 = 102 nM T12475 CY9G1I 67142794 IC50 = 73.8 nM T12475 CED31N 67142818 IC50 = 4.1 nM T12475 C1BV5F 67142820 IC50 > 300 nM T12475 CV0KC5 67142907 IC50 = 20 nM T12475 CMV69X 67142930 IC50 > 100 nM T12475 C3HL4M 67142962 IC50 = 1.5 nM T12475 C86FPN 67142985 IC50 = 3.1 nM T12475 CM83QA 67142995 IC50 = 6.59 nM T12475 C86URV 67142999 IC50 > 300 nM T12475 CIY8A2 67143023 IC50 = 0.17 nM T12475 C5S8LU 67143030 IC50 = 108 nM T12475 CZL0X9 67143054 IC50 = 10 nM T12475 C9FMX1 67143102 IC50 = 103 nM T12475 CBJ8D4 67143119 IC50 = 0.14 nM T12475 CX6CH8 67143135 IC50 = 17.7 nM T12475 CY1J6H 67143374 IC50 = 2 nM T12475 C3Y7PE 67143397 IC50 = 170 nM T12475 CUPF61 67143403 IC50 > 100 nM T12475 CW5EB3 67143407 IC50 = 65.7 nM T12475 C3B4ST 67143413 IC50 = 7.18 nM T12475 CMW0D9 67143415 IC50 > 100 nM T12475 CCY9G3 67143420 IC50 = 2.9 nM T12475 CMTN73 67143432 IC50 = 5.11 nM T12475 C80FIO 67143440 IC50 > 1000 nM T12475 CSP10M 67143454 IC50 > 100 nM T12475 CB20TX 67143468 IC50 > 100 nM T12475 CV7Y5D 67143480 IC50 > 100 nM T12475 C0L8IJ 67143486 IC50 > 100 nM T12475 CT6S8J 67143487 IC50 = 53 nM T12475 C6R7FP 67143490 IC50 = 35.6 nM T12475 C79CEV 67143497 IC50 > 300 nM T12475 CF86DZ 67143505 IC50 = 1.27 nM T12475 CLFT37 67143509 IC50 = 213 nM T12475 C31UWA 67143514 IC50 = 80.3 nM T12475 C76SZF 67143518 IC50 = 0.91 nM T12475 C20HLF 67143534 IC50 > 10 nM T12475 CJ8G7C 67143547 IC50 = 1.16 nM T12475 C3SQV9 67143567 IC50 = 75.6 nM T12475 C6YVM4 67143570 IC50 = 1.42 nM T12475 CI5NP9 67143574 IC50 > 300 nM T12475 CY6ON9 67143587 IC50 > 100 nM T12475 CCP09D 67143598 IC50 = 3.8 nM T12475 CX78QJ 67143604 IC50 > 100 nM T12475 CD3LJ1 67143607 IC50 > 100 nM T12475 C4IWB0 67143612 IC50 = 1.95 nM T12475 C1JZY5 67143613 IC50 = 1.07 nM T12475 C5C1UQ 67143618 IC50 = 0.6 nM T12475 C5N2WJ 67143621 IC50 = 0.39 nM T12475 CU1P3E 67143625 IC50 > 100 nM T12475 C2M0JN 67143633 IC50 = 28.1 nM T12475 C34IEY 67143674 IC50 = 36.9 nM T12475 CP5N1H 67143679 IC50 = 34.2 nM T12475 C7D1XC 67143703 IC50 > 300 nM T12475 C39RJG 67143710 IC50 = 0.32 nM T12475 C2Y3HU 67143715 IC50 = 5 nM T12475 CN2DH4 67143723 IC50 = 42 nM T12475 CE7HU1 67143737 IC50 > 1000 nM T12475 CW20JB 67143740 IC50 > 100 nM T12475 CGA19S 67143743 IC50 = 65.5 nM T12475 C4K5GT 67143746 IC50 > 1000 nM T12475 CC82KM 67143749 IC50 = 35.3 nM T12475 CK4V3D 67143752 IC50 > 100 nM T12475 CZ7I8J 67143755 IC50 = 340 nM T12475 C21IZR 67143761 IC50 = 146 nM T12475 CMZ9N2 67143773 IC50 = 0.39 nM T12475 C02HRB 67143780 IC50 = 0.16 nM T12475 C02RIM 67143786 IC50 > 100 nM T12475 C9EV0T 67143804 IC50 = 1.1 nM T12475 CTZ6A8 67143815 IC50 = 18.2 nM T12475 C48FKB 67143832 IC50 > 1000 nM T12475 CJT9G1 67144077 IC50 > 100 nM T12475 CKZ48L 67144083 IC50 > 100 nM T12475 C5JH9R 67144085 IC50 = 13.3 nM T12475 C6CNL1 67144149 IC50 > 100 nM T12475 CBZ25R 67144162 IC50 = 51.2 nM T12475 CRFL68 67144164 IC50 = 0.31 nM T12475 C9NJI5 67144307 IC50 = 13.9 nM T12475 C19FLN 67144324 IC50 > 100 nM T12475 CW83QO 67144335 IC50 = 115 nM T12475 C1O3TU 67144350 IC50 > 100 nM T12475 CE9PQ1 67144353 IC50 = 0.38 nM T12475 CQX04C 67144367 IC50 = 129 nM T12475 C32UGY 67144370 IC50 = 1.7 nM T12475 C5AHC0 67144393 IC50 > 100 nM T12475 CH97UR 67144408 IC50 = 14.1 nM T12475 CXUF56 67144409 IC50 = 14.2 nM T12475 C6V0NW 67144450 IC50 = 6.8 nM T12475 CY7GO4 67144463 IC50 > 100 nM T12475 CTW73N 67144466 IC50 = 2 nM T12475 C9M7FY 67144478 IC50 = 48.6 nM T12475 CK0SJ1 67144486 IC50 = 65.6 nM T12475 C4FLI9 67144496 IC50 = 8.94 nM T12475 C0X3ZK 67144499 IC50 > 100 nM T12475 CZ6J9U 67144508 IC50 > 100 nM T12475 CJW8A3 67144509 IC50 = 14.8 nM T12475 C2KAZ7 67144531 IC50 = 61 nM T12475 CJH63V 67144582 IC50 = 24.3 nM T12475 CH3WA2 67144628 IC50 > 100 nM T12475 CK3AM4 67144641 IC50 > 1000 nM T12475 CERB89 67144646 IC50 = 7.01 nM T12475 C38GZV 70691201 IC50 = 7.41 nM T12475 CF2X7B 70691931 IC50 = 15.73 nM T12475 CA5Y8U 70697569 IC50 = 110 nM T12475 C5HMI4 70697644 IC50 = 1.36 nM T12475 C2C9DQ 71449058 IC50 = 5.9 nM T12475 CO8Z9S 71459935 Ki = 2.3 nM T12475 CRY8H4 73348538 IC50 = 8.1 nM T12475 CE79LV 73350212 IC50 = 2.01 nM T12475 C49TQS 73351705 IC50 = 2.11 nM T12475 CU0FW3 73356168 IC50 = 3.3 nM T12475 CGR2B3 76335205 IC50 = 0.5 nM T12475 CKDI52 86272223 IC50 = 4210 nM T12475 C7MFW6 86274853 IC50 = 107 nM T12475 C8EFI5 86275342 IC50 = 3.3 nM T12475 C2L9ZS 86275573 IC50 = 5.5 nM T12475 C97SBQ 87285473 IC50 = 27.9 nM T12475 C5NCO3 87285476 IC50 = 0.95 nM T12475 CI6PE1 87285492 IC50 > 300 nM T12475 CNO67R 87285495 IC50 = 217 nM T12475 CK1DN5 87285512 IC50 > 100 nM T12475 CUNS01 87285521 IC50 = 2.57 nM T12475 CSM9N5 87285550 IC50 = 1.2 nM T12475 CO7CA1 87285554 IC50 = 0.39 nM T12475 CQ6UI4 87285560 IC50 > 300 nM T12475 CJU96K 87285565 IC50 = 250 nM T12475 CCR80U 87285570 IC50 = 1.1 nM T12475 CHU98Q 87285576 IC50 > 300 nM T12475 COBI47 87285668 IC50 = 62 nM T12475 CV0QU9 87285708 IC50 = 0.68 nM T12475 C62EPN 87285732 IC50 = 554 nM T12475 CL41WQ 87285735 IC50 > 300 nM T12475 CVP96T 87285767 IC50 = 122 nM T12475 C89PNJ 87285768 IC50 = 0.44 nM T12475 C2GM5X 87285770 IC50 = 184 nM T12475 CH4X5I 118074127 IC50 = 0.23 nM T12475 C49WVD 127036617 IC50 = 588.84 nM T12475 CH1LC4 127036774 IC50 = 724.44 nM T12475 C23MYH 127037454 IC50 = 549.54 nM T12475 C7ZXU0 138978203 Ki = 38 nM T12475 CSUK35 138978204 Ki = 13.8 nM T12475 CHM4L0 138978207 Ki = 395 nM T12475 CZU15V 145948856 IC50 = 281.84 nM T12475 CC5N4A 145948911 IC50 = 407.38 nM T12475 C8IQ4K 145948913 IC50 = 190.55 nM T12475 CF2LM3 145949379 IC50 = 69.1 nM T12475 C4JD8O 145949399 IC50 = 9 nM T12475 CA29XU 145949496 IC50 = 6.3 nM T12475 CDYS96 145949556 IC50 = 73.3 nM T12475 CMA4P8 145950097 IC50 = 46 nM T12475 CQHB07 145950534 IC50 = 144 nM T12475 CK5OS6 145950547 IC50 > 1000 nM T12475 CA6U8B 145951481 IC50 = 45 nM T12475 CT29AE 145951933 IC50 > 100 nM T12475 C8V1OS 145952094 IC50 = 5.4 nM T12475 CFJ06I 145952400 IC50 = 142 nM T12475 C0HG7D 145952498 IC50 = 65.2 nM T12475 C7YJ2Q 145952802 IC50 = 7.5 nM T12475 CW23GF 145953172 IC50 = 1.21 nM T12475 CLV0J7 145953549 IC50 = 15.2 nM T12475 CI7HC0 145954246 IC50 = 0.38 nM T12475 CF05AH 145954419 IC50 = 3.03 nM T12475 CD4CN3 145954439 IC50 = 22 nM T12475 CBC86M 145954593 IC50 = 62.3 nM T12475 C5ZK9S 145955182 IC50 = 17.2 nM T12475 CT2IO8 145955260 IC50 = 1682 nM T12475 C23EQA 145955571 IC50 = 0.33 nM T12475 CEP1U3 145955844 IC50 = 0.74 nM T12475 CU0V3R 145956692 IC50 = 89 nM T12475 CX0N9S 145957253 IC50 = 38.5 nM T12475 CDHK42 145957335 IC50 = 49.5 nM T12475 C6ZCM0 145957339 IC50 = 16 nM T12475 CD9N2O 145957402 IC50 > 1000 nM T12475 CHSR47 145957680 IC50 = 19.1 nM T12475 C1M3YZ 145957893 IC50 = 6.2 nM T12475 CYSH48 145957953 IC50 = 1.54 nM T12475 CLY84H 145958075 IC50 = 32 nM T12475 CWNG28 145958346 IC50 = 0.29 nM T12475 CT58YA 145958486 IC50 = 20.4 nM T12475 C2FD5N 145959547 IC50 = 1066 nM T12475 CT1SB4 145962692 IC50 = 2.3 nM T12475 C5RYZ6 145973124 IC50 = 11.3 nM T12475 C09AFT 145973618 IC50 = 8.4 nM T12475 C2GQ3U 145973813 IC50 = 160 nM T12475 CD0MF8 145980339 Ki = 254 nM T12475 CG98XV 145981421 Ki > 1000 nM T12475 C0HI7Z 145984647 Ki = 410 nM T12475 C1BC8G 145989544 Ki > 1000 nM T12475 CTCI50 145991962 Ki = 104 nM T12475 CA12SD 145992260 Ki = 157 nM T12475 CL08YC 145993478 Ki = 186 nM T12475 CSM51N 155517188 IC50 = 0.69 nM T12475 CA6TV7 155524081 IC50 = 0.11 nM T12475 C5N9EB 155531714 IC50 = 1.63 nM T12475 C87ZKL 155538326 IC50 = 226 nM T12475 C1W2AQ 155559612 IC50 = 7.1 nM T12475 CFK31W 155569451 IC50 = 2.4 nM T12475 CO09MC 45263736 Ki = 0.36 nM T12475 D00HNG 9957278 Ki = 6 nM T12475 D00JYL 16221495 IC50 = 0.81 nM T12475 D00TSY 16156517 IC50 = 3.162 nM T12475 D01DBW 16221494 IC50 = 0.31 nM T12475 D02NCO 9874838 Ki = 0.1 nM T12475 D03JDY 16221150 IC50 = 4.6 nM T12475 D03YHT 16221496 IC50 = 0.87 nM T12475 D04BVX 16221556 IC50 = 0.83 nM T12475 D04HPP 16221613 IC50 = 39 nM T12475 D04TDF 16156445 IC50 = 0.912 nM T12475 D05ELQ 16221211 IC50 = 1.2 nM T12475 D05UTO 16155218 IC50 = 3.46 nM T12475 D07DPW 16221212 IC50 = 3 nM T12475 D07XFF 16156634 IC50 = 0.8511 nM T12475 D08XDH 16155593 IC50 = 1.072 nM T12475 D09UXO 16155098 IC50 = 1.69 nM T12475 D0B6LL 16155587 IC50 = 0.6 nM T12475 D0C0HP 10231401 IC50 = 7.2 nM T12475 D0C2JJ 16155709 IC50 = 0.51 nM T12475 D0C7LY 11496610 IC50 = 12 nM T12475 D0G6IX 16221557 IC50 = 13 nM T12475 D0I9JL 16221433 IC50 = 1.2 nM T12475 D0K1AT 16221434 IC50 = 25 nM T12475 D0K2MC 16221267 IC50 = 0.6 nM T12475 D0K8AP 16202050 IC50 = 3.16 nM T12475 D0KA9Y 16221266 IC50 = 0.8 nM T12475 D0L8WJ 16156699 IC50 = 0.8128 nM T12475 D0O5VA 9833530 IC50 = 1.9 nM T12475 D0R9JG 16155654 IC50 = 2.68 nM T12475 D0RB5Z 16138575 IC50 = 2.2 nM T12475 D0W5JT 16221328 IC50 = 6.2 nM T12475 D0WG8L 16221379 IC50 = 85 nM T12475 D0X1RZ 16156573 IC50 = 0.88 nM T12475 D0XL0H 16221614 IC50 = 2004 nM T12475 D0Y1WD 16221104 IC50 = 0.73 nM T12475 D0Y2NA 16221329 IC50 = 3815 nM T12475 D0Z5TP 16221151 IC50 = 6.9 nM T89859 CH03PR 9866186 IC50 = 2500 nM T89859 CWJ2N6 23577107 IC50 = 8000 nM T89859 CJ7UP5 23577110 IC50 = 500 nM T89859 CW2H8L 25023779 IC50 = 1000 nM T97141 D04OSE 4485 IC50 = 2020 nM T97141 D03KKR 3547 IC50 = 3600 nM T97141 D08ZPO 448043 Ki = 10100 nM T97141 D0E3TC 44259 IC50 = 10 nM T97141 D0P1JI 312145 IC50 = 1900 nM T97141 C8Z1FA 1960 Ki = 7400 nM T97141 CZM9B7 2404 IC50 = 3700 nM T97141 CA47TS 3546 Ki = 150000 nM T97141 C95GCZ 3568 IC50 = 17800 nM T97141 CWT4N9 4216 Ki = 300 nM T97141 CKEB49 5681 Ki = 110000 nM T97141 CFD0V9 132904 IC50 = 10000 nM T97141 C0MF7L 476293 IC50 = 200 nM T97141 C18WEB 490561 Ki = 17 nM T97141 CAVO87 686075 IC50 > 100000 nM T97141 C63WLU 939124 IC50 > 100000 nM T97141 CYF3U0 5327849 IC50 = 1600 nM T97141 CG8X2O 5327850 IC50 = 30 nM T97141 CLQ16T 5327851 IC50 = 390 nM T97141 CTMF93 5327852 IC50 = 220 nM T97141 CPQ0M3 5327853 IC50 = 310 nM T97141 CF3D5E 5327854 IC50 = 250 nM T97141 C75HPA 5327855 IC50 = 18 nM T97141 CJZ87B 5327856 IC50 = 5500 nM T97141 CJED26 5327858 IC50 = 55 nM T97141 CE13YF 5327859 IC50 = 49 nM T97141 CLP17B 5327860 IC50 = 180 nM T97141 C6ISZ2 5327862 IC50 = 120 nM T97141 C9D5JI 9879020 IC50 = 690 nM T97141 CRO5D3 9912410 IC50 = 25 nM T97141 COW68T 11605551 IC50 = 17800 nM T97141 C38FDZ 16760660 IC50 = 10 ug.mL-1 T97141 CXF7G4 21216838 IC50 = 32 nM T97141 CY8L7E 24896769 IC50 > 10000 nM T97141 C8QY9B 44225231 IC50 = 23300 nM T97141 CN1O5R 44225232 IC50 = 33300 nM T97141 C15HTU 44225473 IC50 = 13300 nM T97141 CC5BU8 44225474 IC50 = 31300 nM T97141 C74KYR 44225475 IC50 = 41300 nM T97141 CC0WU4 44225476 IC50 = 3300350.01 nM T97141 C5WY3D 44225477 IC50 = 9803925.45 nM T97141 CAHC93 44225478 IC50 = 15200 nM T97141 C7GY0A 44225710 IC50 = 9800 nM T97141 C8EOZ6 44225711 IC50 = 5208348.07 nM T97141 CZG91W 44225712 IC50 = 29200 nM T97141 CUEZ83 44225713 IC50 = 5100 nM T97141 CK29SZ 44225714 IC50 = 7400 nM T97141 CG0JQ7 44225715 IC50 = 24390460.5 nM T97141 C7OV0A 44370409 IC50 = 9200 nM T97141 COT05F 44450721 IC50 = 3700 nM T97141 CNX84R 44817010 IC50 = 900 nM T97141 C0DRX5 50898538 IC50 = 36000 nM T97141 C67VCL 52947006 IC50 = 51000 nM T97141 CX13OD 53316491 IC50 = 23600 nM T97141 C1NLD5 53317828 IC50 = 25100 nM T97141 CI6A9B 53324357 IC50 = 8700 nM T97141 CV63UL 67240318 IC50 > 10000 nM T97141 CSE6Z5 71463101 EC50 > 20000 nM T97141 CDJY72 71568837 IC50 = 4000 nM T97141 C8CAG7 71578921 IC50 > 10000 nM T97141 C0DL3F 72698602 IC50 = 15.63 nM T97141 C4U5NV 73442760 IC50 = 1000000 nM T97141 CCS27Y 101899357 IC50 = 9100 nM T97141 C8PAX5 122190865 IC50 = 18200 nM T97141 CSR85E 122190866 IC50 = 10204224.39 nM T97141 C65DTF 122190919 IC50 = 7300 nM T97141 CAR4K7 122190920 IC50 = 4300 nM T97141 CG8K3C 122190921 IC50 = 4210 nM T97141 CUIT13 122190922 IC50 = 2140 nM T97141 C3Q1NC 122190923 IC50 = 2040 nM T97141 CUZ19F 122190924 IC50 = 2040 nM T97141 CH9I4J 122190925 IC50 = 4370 nM T97141 C94CZL 122190926 IC50 = 3670 nM T97141 C7NV1J 122190927 IC50 = 10800 nM T97141 CYK86O 122190928 IC50 = 11100 nM T97141 CDSA68 122190929 IC50 = 13300 nM T97141 CA93QX 122190930 IC50 = 4700 nM T97141 C8PLK2 122190931 IC50 = 5900 nM T97141 CH4BC9 122190932 IC50 = 2170 nM T97141 CA5YT7 122190933 IC50 = 2100 nM T97141 CG1X7I 122190934 IC50 = 3040 nM T97141 C41VCR 122190935 IC50 = 7370 nM T97141 CG8BQ5 122190936 IC50 = 3670 nM T97141 CTF1S2 122190937 IC50 > 100000 nM T97141 C2MD1Q 155513187 IC50 > 10000 nM T97141 D01SLS 4217 Ki = 3800 nM T97141 D03DYT 3035817 Ki = 20 nM T97141 D07OAK 3500 IC50 = 120 nM T97141 D08JPU 3501 IC50 = 5800 nM T97141 D09FFE 449241 Ki = 28300 nM T97141 D0O0VZ 667639 IC50 = 12000 nM T97141 D0T3PW 5281672 Ki = 1700 nM T66686 CRZ50H 10838633 IC50 > 10000000 nM T66686 CVE50F 44347762 IC50 > 10000000 nM T66686 C7XYS9 44347952 IC50 > 10000000 nM T66686 CE84VF 44347974 IC50 > 10000000 nM T78932 D03ZBT 11626560 IC50 = 1269 nM T78932 D04LKS 25126798 IC50 = 0.4 nM T78932 D0EG1I 9926791 Ki = 4.39 nM T78932 D0Y7IC 44205240 IC50 = 8.7 nM T78932 D00RYA 16750271 IC50 = 230 nM T78932 D02TUL 118115473 IC50 > 10000 nM T78932 D03HUX 49792852 IC50 > 10000 nM T78932 D03LWG 53235510 IC50 = 3303 nM T78932 D04QWQ 59422203 IC50 = 11 nM T78932 D05PCM 78323835 IC50 > 200000 nM T78932 D05PZB 135398495 IC50 = 1 nM T78932 D06EIC 57928403 IC50 = 4.8 nM T78932 D07EHV 44814409 IC50 > 10000 nM T78932 D07HPJ 11476171 IC50 > 10000 nM T78932 D07JAG 58557659 IC50 = 4690 nM T78932 D0D8KQ 25127112 IC50 = 116 nM T78932 D0DK5X 135567296 IC50 = 29.7 nM T78932 D0DK8X 50922691 IC50 = 66 nM T78932 D0E3TC 44259 IC50 = 0.351 nM T78932 D0G8BM 16722836 IC50 = 150 nM T78932 D0PN8H 46216796 IC50 = 50 nM T78932 D0S1XX 134821691 Ki = 0.02 nM T78932 D0SG7B 49831257 IC50 = 116 nM T78932 CU68FI 78893 Ki = 3100 nM T78932 C6ZB4U 790291 Ki = 1200 nM T78932 CGQM48 869412 Ki = 790 nM T78932 C0XL5P 951379 Ki > 3500 nM T78932 C7ZUW6 1246120 Ki = 540 nM T78932 CI1B7L 1247281 Ki > 3500 nM T78932 C3F0GS 3120536 Ki = 230 nM T78932 CD67OL 4250390 Ki = 2400 nM T78932 C6SNL5 4393251 Ki = 1100 nM T78932 CK6L3O 5121684 Ki = 1100 nM T78932 CUJR40 10062694 EC50 > 2000 nM T78932 CO70CQ 10107882 IC50 = 937 nM T78932 CBOP58 11293798 Ki > 10000 nM T78932 C26BZX 11362471 Ki > 10000 nM T78932 CWXB93 11397177 Ki > 10000 nM T78932 CTG83F 11539329 Ki > 1900 nM T78932 CMIL86 11590363 Ki > 1900 nM T78932 C9T6SC 11640926 Ki > 1900 nM T78932 C75SGK 12997800 IC50 = 7 nM T78932 CFPW41 16007116 Ki > 1900 nM T78932 CKR57M 16086104 IC50 = 2730 nM T78932 C16NRY 16086114 IC50 = 1830 nM T78932 CSE35D 16739464 IC50 = 1500 nM T78932 C20OFQ 16739508 IC50 = 710 nM T78932 CCP56J 16739905 IC50 = 41 nM T78932 CQ64XI 16739921 IC50 = 33 nM T78932 CM3UF8 16739935 IC50 = 590 nM T78932 CFEP56 16739948 IC50 = 65 nM T78932 C23KZR 16739951 IC50 = 5900 nM T78932 C9OQ1G 16750272 IC50 = 670 nM T78932 CW2SY5 16750291 IC50 = 32 nM T78932 CIX7U2 16750304 IC50 = 120 nM T78932 C6A3XS 16750306 IC50 = 47 nM T78932 CB2TK1 16750327 IC50 = 310 nM T78932 CH4O1C 16750328 IC50 = 630 nM T78932 C90MJD 16750331 IC50 = 950 nM T78932 C6UAZ0 20820292 IC50 = 360 nM T78932 CE7K3W 23532567 IC50 > 10000 nM T78932 CUY98W 23585560 IC50 = 66 nM T78932 CD0R9O 24699546 Ki = 380 nM T78932 C7YG1N 24759534 IC50 = 75 nM T78932 CLBP72 24798571 IC50 = 519 nM T78932 CX1U4S 24800423 IC50 = 3400 nM T78932 C4T0DG 24800602 IC50 > 10000 nM T78932 CH3ZG7 24800604 IC50 > 10000 nM T78932 CBA02Y 24800776 IC50 = 1400 nM T78932 C3UFG1 24801129 IC50 = 150 nM T78932 CVR8S1 24801650 IC50 = 640 nM T78932 CWV98O 24899557 IC50 = 1500 nM T78932 C0JYA9 25123154 IC50 = 2900 nM T78932 C56JVD 25123155 IC50 = 640 nM T78932 CZM6Q2 25123472 IC50 = 340 nM T78932 C3IA7V 25123474 IC50 > 10000 nM T78932 C6V4NB 25123475 IC50 = 1400 nM T78932 CFK89A 25123806 IC50 = 520 nM T78932 C3RMN9 25123807 IC50 = 2200 nM T78932 C5GO3T 25123808 IC50 = 7130 nM T78932 C4WFL0 25128110 IC50 = 640 nM T78932 COV8Z0 25143021 IC50 > 10000 nM T78932 CI0E2L 25154395 IC50 = 30 nM T78932 CL1W5D 25154436 IC50 = 72 nM T78932 C0ZXH7 25236808 Ki = 230 nM T78932 CT7X8Y 27700054 Ki > 3500 nM T78932 C3VRO9 44557921 IC50 > 10000 nM T78932 C5YL2S 44570390 IC50 = 280 nM T78932 C6QT0J 44622837 IC50 > 1000 nM T78932 CY3HW5 46224684 IC50 = 10000 nM T78932 C1S4LH 46398810 IC50 = 384 nM T78932 C35AIH 46865430 IC50 = 120 nM T78932 C2EK4B 46865431 IC50 = 200 nM T78932 CMZ0R3 46865529 IC50 = 94 nM T78932 C3B2NL 46865530 IC50 = 86 nM T78932 CLS29B 46872626 IC50 > 10000 nM T78932 C5NZ8R 46880686 IC50 = 3600 nM T78932 CZ79VE 46880687 IC50 = 110 nM T78932 C0YNH6 46880737 IC50 = 63 nM T78932 CGO7C5 46880738 IC50 = 310 nM T78932 C75ZTG 46880739 IC50 = 730 nM T78932 C9T7WL 46880784 IC50 = 300 nM T78932 CSV4G2 46880785 IC50 = 97 nM T78932 C9MW2L 46885052 IC50 > 10000 nM T78932 C69HUW 46885053 IC50 > 10000 nM T78932 CASL67 46885231 IC50 = 4200 nM T78932 CEU6O4 46885232 IC50 = 9300 nM T78932 CE27LI 46885233 IC50 = 330 nM T78932 CB8LN4 46885234 IC50 = 439 nM T78932 CMX7U6 46885289 IC50 = 520 nM T78932 CB1ZN5 46885290 IC50 = 120 nM T78932 C2O8RZ 46886323 IC50 > 1000 nM T78932 CT7EY8 49817363 IC50 = 4333 nM T78932 C9L3XR 49838879 IC50 > 5000 nM T78932 CON2Z1 49839198 Ki = 11.1 nM T78932 CB34CO 49839441 Ki = 19 nM T78932 C2DGY0 49839445 Ki > 3500 nM T78932 C06MKW 49839561 Ki = 4.8 nM T78932 CD8TK0 49839914 Ki = 9.5 nM T78932 CRA74I 49842779 IC50 > 10000 nM T78932 CF91RS 49843531 IC50 > 10000 nM T78932 C7A6IZ 49850211 IC50 = 4800 nM T78932 CK4LJ5 49856703 Ki = 3500 nM T78932 CA0WR3 50914031 IC50 = 150 nM T78932 CQE9D1 50925411 IC50 = 1691 nM T78932 C2Y6QS 50938552 IC50 > 10000 nM T78932 C20VEP 50994284 IC50 > 10000 nM T78932 CI1L0M 50994285 IC50 > 10000 nM T78932 C7ZWT8 50994286 IC50 > 10000 nM T78932 C6VNE1 50994366 IC50 = 5040 nM T78932 CSEZ73 50994367 IC50 > 10000 nM T78932 C9NYP4 51036677 IC50 > 10000 nM T78932 C4WRY3 51037112 IC50 > 10000 nM T78932 CRI28Z 51037948 IC50 > 10000 nM T78932 CA9DE6 52941228 IC50 = 760 nM T78932 C1T5EH 52942437 IC50 = 690 nM T78932 CEPS91 52943663 IC50 = 70 nM T78932 C2IQ5B 52943672 IC50 = 6040 nM T78932 CW5LG6 52943677 IC50 > 10000 nM T78932 CUT89J 52944095 IC50 > 10000 nM T78932 CSY3F8 52944096 IC50 > 10000 nM T78932 CF8VA5 52944440 IC50 > 10000 nM T78932 CTN0C3 52944839 IC50 = 1720 nM T78932 CT2U3E 52947304 IC50 = 70 nM T78932 CPEO70 52947328 IC50 > 10000 nM T78932 CQY9D0 52948526 IC50 = 42 nM T78932 C8TC3P 52948550 IC50 = 70 nM T78932 CIM43G 52948562 IC50 = 300 nM T78932 CY4NI1 52950144 IC50 > 10000 nM T78932 CZ0BV7 53320342 IC50 > 10000 nM T78932 C2W9OA 53324451 IC50 = 4400 nM T78932 CZKQ72 53341161 Ki = 234 nM T78932 CB83XH 53341368 Ki = 250 nM T78932 CGP23R 53341457 Ki = 4.7 nM T78932 C95JTI 53373594 Ki = 0.6 nM T78932 CM12OQ 53475998 Ki = 13 nM T78932 C6W0PN 53476000 Ki = 19 nM T78932 C4G2ST 53476104 Ki = 0.6 nM T78932 C37PHN 53497571 IC50 = 1330 nM T78932 CCF1B3 53497572 IC50 = 266 nM T78932 C1XS2J 54760383 IC50 = 6700 nM T78932 CR9A5O 56834874 IC50 = 4100 nM T78932 C58MSV 56834889 IC50 = 757 nM T78932 CJBL48 56925034 IC50 = 753 nM T78932 CBFR12 56925356 IC50 = 1070 nM T78932 C80DRA 56925357 IC50 = 1990 nM T78932 C0HUN8 56925358 IC50 = 2600 nM T78932 C6Z2EA 56925359 IC50 = 6980 nM T78932 CC1MN2 56925454 IC50 = 5150 nM T78932 C3XC0T 56925455 IC50 = 888 nM T78932 CBW6T3 56925456 IC50 = 202 nM T78932 C8G3NO 56925457 IC50 = 208 nM T78932 CHS19C 56925458 IC50 = 146 nM T78932 CBMO42 56925459 IC50 = 932 nM T78932 CQTD41 56925550 IC50 = 1480 nM T78932 CI9T3S 56925551 IC50 = 2670 nM T78932 CS84ZU 56925552 IC50 = 1550 nM T78932 C9IVD0 56929216 Ki = 6.2 nM T78932 C0BO4X 56934550 Ki = 1.6 nM T78932 CJMB49 56953110 Ki = 0.5 nM T78932 CSO40C 56973425 Ki = 85 nM T78932 CPO2J4 57342178 IC50 = 150 nM T78932 CA93PN 57342180 IC50 = 440 nM T78932 C3KQJ8 57928435 IC50 = 4.8 nM T78932 C8R4FE 57991377 IC50 = 348.3 nM T78932 CD6ZP3 58009815 IC50 = 60 nM T78932 CWU1Y3 58009825 IC50 = 300 nM T78932 C8S6MY 58010054 IC50 = 50 nM T78932 CKA28H 58180521 IC50 = 1.9 nM T78932 C2I5LO 58180525 IC50 = 46 nM T78932 CWXC70 58180596 IC50 = 110 nM T78932 C9N1QB 58180623 IC50 = 220 nM T78932 CSK1U8 58180628 IC50 = 28 nM T78932 C6LT9S 58180630 IC50 = 45 nM T78932 CP81TW 58394456 Ki = 540 nM T78932 C0F3BO 58394783 Ki = 31 nM T78932 CO5TH6 58394820 Ki = 71 nM T78932 C0X7IK 58394837 Ki = 12 nM T78932 C9Q4WD 58394916 Ki = 89 nM T78932 CASI81 58395078 Ki = 0.4 nM T78932 CDK5L1 58395223 Ki = 20 nM T78932 CWBM72 58395283 Ki = 1.7 nM T78932 C9MIL7 58450666 IC50 = 774 nM T78932 CB42EF 58557147 IC50 = 530 nM T78932 CZ3TG1 59375154 IC50 > 2000 nM T78932 CXJ63M 59603829 IC50 = 92 nM T78932 CQEU96 59603842 IC50 = 52 nM T78932 C8UMJ2 59617909 Ki = 1500 nM T78932 C51LST 59617917 Ki = 13.5 nM T78932 CDMO01 59617921 Ki = 840 nM T78932 CUNY05 59617942 Ki > 3500 nM T78932 CY7V3I 59617971 Ki = 250 nM T78932 CNOE97 59618008 Ki = 7.8 nM T78932 CM6B3E 59618010 Ki = 94 nM T78932 C2DWY5 59618025 Ki = 5.1 nM T78932 CQCG48 59618036 Ki = 1200 nM T78932 CHS43W 59618040 Ki = 7.6 nM T78932 CJ5GF1 59618081 Ki > 3500 nM T78932 C3Q1NR 59618098 Ki = 8.5 nM T78932 COMD30 59618112 Ki = 4.4 nM T78932 CT12JO 59618117 Ki = 140 nM T78932 CRM8E5 59618118 Ki = 11.4 nM T78932 C42OZL 59618123 Ki = 14 nM T78932 C2GU4R 59618132 Ki = 3.2 nM T78932 COI26N 59618146 Ki = 2800 nM T78932 CR5GJ4 59618147 Ki = 1500 nM T78932 C9GB1C 59618160 Ki = 1200 nM T78932 CR9F7D 59618164 Ki = 96 nM T78932 C7XWE2 59618171 Ki = 74 nM T78932 C3WEG9 59618205 Ki = 7.8 nM T78932 CNZ10K 59618273 Ki = 1.8 nM T78932 C2EIA3 59618285 Ki = 29 nM T78932 C1ZKR9 59618313 Ki = 930 nM T78932 CHFN86 59618317 Ki = 3 nM T78932 C10HYQ 59618327 Ki = 22.2 nM T78932 C7ET9U 59618334 Ki = 60.8 nM T78932 COY0T1 59618339 Ki = 5.4 nM T78932 C61LWQ 59618347 Ki = 1 nM T78932 CA67ON 59618368 Ki = 2.5 nM T78932 C0X9SW 59618378 Ki = 7.1 nM T78932 C26BNV 59618424 Ki = 2000 nM T78932 C3B7CU 59618428 Ki = 10 nM T78932 CBH83T 59618445 Ki = 240 nM T78932 C7WI0Y 59618449 Ki = 3.1 nM T78932 C3HC4P 59618462 Ki = 240 nM T78932 CCOP27 59618475 Ki = 30.1 nM T78932 CF2U0A 59618498 Ki = 14.6 nM T78932 COEK07 59618504 Ki = 1.3 nM T78932 CX0FQ2 59618505 Ki = 4.9 nM T78932 C0UYI9 59618511 Ki = 1.4 nM T78932 CG8ET4 59618513 Ki = 64 nM T78932 C7PF3G 59618531 Ki = 35.1 nM T78932 CU04RZ 59618547 Ki = 21.8 nM T78932 CR27IT 59618564 Ki = 1900 nM T78932 CNY59P 60165955 Ki = 4.2 nM T78932 CY3QT8 60165956 Ki = 160 nM T78932 CJ08ZL 66604045 IC50 = 171 nM T78932 CY0I2V 66604274 IC50 = 71 nM T78932 CD0LJ6 66604359 IC50 = 31 nM T78932 CS8HK2 66604394 IC50 = 16 nM T78932 C7U8GC 66604464 IC50 = 201 nM T78932 CXU94O 66604576 IC50 = 179 nM T78932 CE9T0V 66604664 IC50 = 608 nM T78932 C7WO4A 66604791 IC50 = 45 nM T78932 CW53KR 66604810 IC50 = 247 nM T78932 CNW05G 66604855 IC50 = 40 nM T78932 C0JS8O 66604914 IC50 = 2.8 nM T78932 CW9LD1 66604921 IC50 = 129 nM T78932 CTMX20 66605009 IC50 = 70 nM T78932 CP0DB1 66605115 IC50 = 87 nM T78932 CB1WC9 66605298 IC50 = 243 nM T78932 CCWU74 66605322 IC50 = 32 nM T78932 C7Q8ZG 66605359 IC50 = 158 nM T78932 C16TEK 66605475 IC50 = 117 nM T78932 C7MOJ6 66605487 IC50 = 160 nM T78932 CDZA70 66605639 IC50 = 197 nM T78932 C53NBQ 66605756 IC50 = 39 nM T78932 C1HSE0 67035086 IC50 = 1500 nM T78932 CWI6K5 67035106 IC50 > 10000 nM T78932 C38RGB 67035556 IC50 > 10000 nM T78932 CV63UL 67240318 IC50 > 10000 nM T78932 CKMV48 67345882 Ki = 3.4 nM T78932 CFX84K 67352945 Ki = 80 nM T78932 CEF67O 67383086 Ki = 0.3 nM T78932 CLO13H 67383145 Ki = 0.7 nM T78932 C94UAF 67383148 Ki = 3.2 nM T78932 C5D2QA 67383227 Ki = 0.7 nM T78932 C4AE8Z 67383253 Ki = 1.2 nM T78932 CW8Q3F 67383552 Ki = 1 nM T78932 C6UF3T 67383612 Ki = 0.4 nM T78932 CV38SD 67383669 Ki = 5.1 nM T78932 C9WY2P 67383875 Ki = 0.7 nM T78932 CJ2Q1S 67383893 Ki = 0.5 nM T78932 CUK87J 67387753 Ki = 1.7 nM T78932 CZ0O6N 68234726 Ki = 0.5 nM T78932 CA89HR 68235185 Ki = 9.9 nM T78932 C4U1IR 68291322 IC50 = 22 nM T78932 C2P7DB 68291391 IC50 = 52 nM T78932 CRM3S0 68291627 IC50 = 110 nM T78932 C4LKB3 68291752 IC50 = 2 nM T78932 CQ49HB 68291755 IC50 = 34 nM T78932 CXI4L1 68291797 IC50 = 110 nM T78932 C8T5VB 68291830 IC50 = 97 nM T78932 CPRW18 68291866 IC50 = 118 nM T78932 C6UWI3 68291981 IC50 = 110 nM T78932 CYN89R 68292156 IC50 = 30 nM T78932 C76EZC 68292170 IC50 = 79 nM T78932 CGA0W6 68292183 IC50 = 6 nM T78932 C93LZT 68292196 IC50 = 400 nM T78932 C8I7GC 68293638 IC50 > 10000 nM T78932 CD56XK 68293660 IC50 > 10000 nM T78932 CK6N8J 68686405 Ki = 10.9 nM T78932 COQ9D2 68692728 Ki = 3.4 nM T78932 C6M7ZH 68758088 Ki = 3.3 nM T78932 C5DGR9 69036886 IC50 = 10000 nM T78932 CVH5M3 69671224 Ki = 1.3 nM T78932 CW4JA3 70823673 Ki = 9.1 nM T78932 CQ2F8J 70824464 Ki = 170 nM T78932 C3JLU7 70824497 Ki = 15 nM T78932 CJH94D 71062030 IC50 = 130 nM T78932 COD6B2 71222450 Ki = 0.6 nM T78932 C7Y2LB 71230234 Ki = 20 nM T78932 CKT60L 71455860 Ki > 1900 nM T78932 CCN01X 71547862 IC50 > 10000 nM T78932 CCG31P 71682467 Ki = 10.3 nM T78932 CF08MS 71682929 Ki = 1.6 nM T78932 C5QK6S 71727668 IC50 = 0.6 nM T78932 C1N7LQ 72202249 IC50 = 3 nM T78932 C6THF4 72374600 Ki = 18 nM T78932 CNJ03L 72375990 Ki > 3500 nM T78932 C5R0WV 72375991 Ki > 3500 nM T78932 CVUL48 72375992 Ki = 900 nM T78932 CO8KW2 72375993 Ki = 2800 nM T78932 CN0I2W 72375994 Ki > 3500 nM T78932 C1XD7U 72375995 Ki = 3200 nM T78932 C8BJ4U 72375996 Ki > 3500 nM T78932 C7XFW2 72375997 Ki > 3500 nM T78932 CJB95D 72375998 Ki > 3500 nM T78932 CS5V9L 72376089 Ki > 3500 nM T78932 C37GPL 72376090 Ki > 3500 nM T78932 C9U3WO 72376091 Ki > 3500 nM T78932 CK7F6U 72700776 Ki = 11 nM T78932 CRAW59 73349195 Ki = 100 nM T78932 CL4SD8 73355260 Ki > 3500 nM T78932 C4KF0H 75201716 IC50 = 62 nM T78932 C7M4FR 75201717 IC50 = 0.95 nM T78932 C0OJ7W 75201718 IC50 = 190 nM T78932 C2S0CO 75201720 IC50 = 19 nM T78932 C5S2HO 75201785 IC50 = 69 nM T78932 C4U5MR 75201786 IC50 = 15 nM T78932 C6S2ZO 75201851 IC50 = 630 nM T78932 CO0BQ5 76310565 IC50 = 5827 nM T78932 C6ZAB2 76310566 IC50 > 10000 nM T78932 C0F6VU 76310567 IC50 > 10000 nM T78932 CDO38G 76310568 IC50 > 10000 nM T78932 CL42BQ 76310569 IC50 > 10000 nM T78932 CWI1Q4 76310570 IC50 = 11927 nM T78932 C7SXJ1 76314208 IC50 > 10000 nM T78932 CSDI71 76314209 IC50 = 995 nM T78932 CXF1I3 76317774 IC50 > 10000 nM T78932 CY79VS 76317775 IC50 > 10000 nM T78932 CNK2I1 76317776 IC50 = 7368 nM T78932 CS02NA 76317777 IC50 = 5104 nM T78932 CAHW32 76317778 IC50 > 10000 nM T78932 C2SMK1 76321491 IC50 > 10000 nM T78932 C2DSX7 76321492 IC50 > 10000 nM T78932 CXA4O1 76325093 IC50 > 10000 nM T78932 C8GK0H 76328659 IC50 > 10000 nM T78932 CJN89E 76332335 IC50 > 10000 nM T78932 CW1QK4 76332336 IC50 > 10000 nM T78932 C2P1MX 76332338 IC50 > 10000 nM T78932 CB4KQ7 76335967 IC50 > 10000 nM T78932 C84PFQ 76335968 IC50 = 9844 nM T78932 CW1HQ9 76370451 IC50 = 4.8 nM T78932 CD6Y1F 78320046 IC50 > 200000 nM T78932 CW08SU 78320048 IC50 > 200000 nM T78932 CWI93D 78323836 IC50 > 200000 nM T78932 C5UK9L 78323837 IC50 > 200000 nM T78932 CQ3EJ1 78324132 IC50 > 200000 nM T78932 C7VOX0 78324136 IC50 > 200000 nM T78932 CA2Y8L 78324435 IC50 > 200000 nM T78932 C4I7WD 78324744 IC50 > 200000 nM T78932 CPG3A5 86302574 IC50 > 30000 nM T78932 C96EDF 86660048 IC50 = 650 nM T78932 CC8I0M 86707711 IC50 = 25 nM T78932 CW4Z2F 89470642 IC50 = 1.2 nM T78932 CBRF87 89470690 IC50 = 3 nM T78932 C7B8OH 89470730 IC50 = 0.4 nM T78932 CDQ8C6 89471114 IC50 = 2 nM T78932 C4G5LP 89471136 IC50 = 2.9 nM T78932 CU6J4F 89498235 Ki = 0.6 nM T78932 C1HW4B 89735655 IC50 = 10000 nM T78932 C13GOX 89775209 IC50 = 33 nM T78932 C3N6RU 89775221 IC50 = 5.5 nM T78932 CT8G2E 90135056 IC50 = 120 nM T78932 CXZ3L7 90135672 IC50 = 40 nM T78932 CG5P9A 90153688 IC50 = 0.92 nM T78932 CKY9T6 90153726 IC50 = 570 nM T78932 C0C7FO 90153735 IC50 = 23 nM T78932 CRC2D0 90153737 IC50 = 100 nM T78932 CV6H7R 90153809 IC50 = 12 nM T78932 CLU1E6 90153817 IC50 = 87 nM T78932 CFC48T 90153820 IC50 = 300 nM T78932 C1FUQ2 90153821 IC50 = 79 nM T78932 CTSV65 90153949 IC50 > 10000 nM T78932 C04KWP 90154028 IC50 = 170 nM T78932 CUR62C 90154140 IC50 = 11 nM T78932 CV64KY 90183363 Ki > 1000 nM T78932 CTV52A 90367281 IC50 = 13 nM T78932 CFB75T 90479825 IC50 = 5 nM T78932 CY0UC4 90645194 IC50 > 10000 nM T78932 C7EXH8 91755097 IC50 = 34 nM T78932 C37IZB 91755098 IC50 = 180 nM T78932 C7UAK5 91809175 Ki = 0.086 nM T78932 C8RG6H 91827514 IC50 = 690 nM T78932 C64SIO 92042864 IC50 > 10000 nM T78932 C9BL4M 92045136 IC50 = 28000 nM T78932 CXU1Z2 101043725 IC50 = 970 nM T78932 CRI0S4 101891768 Ki > 1000 nM T78932 CM2C3W 105539869 IC50 = 30 nM T78932 C3ECY5 117625437 IC50 = 0.55 nM T78932 CZC84D 117769161 IC50 = 14 nM T78932 CE7BZ8 117769174 IC50 = 190 nM T78932 CBJ07Q 117769217 IC50 = 46 nM T78932 CXHQ08 117769229 IC50 = 12 nM T78932 CS9WO4 117769234 IC50 = 7.9 nM T78932 C61VXQ 117769241 IC50 = 10 nM T78932 C1SA9I 117769244 IC50 = 27 nM T78932 C0VY7C 117769271 IC50 = 21 nM T78932 C6O9BT 117769272 IC50 = 55 nM T78932 CSR9B0 117769289 IC50 = 30 nM T78932 C2M9CR 117769307 IC50 = 59 nM T78932 C7FWS3 117769309 IC50 = 8.6 nM T78932 CYWV32 117769339 IC50 = 47 nM T78932 CZV35K 117769346 IC50 = 14 nM T78932 C5V6RG 117769349 IC50 = 44 nM T78932 C4O1PX 117769362 IC50 = 22 nM T78932 CPV4C8 117769365 IC50 = 9.2 nM T78932 CP3MC5 117769379 IC50 = 15 nM T78932 C8V6LG 117769392 IC50 = 29 nM T78932 C2NBZ8 117769396 IC50 = 20 nM T78932 COV59Y 117769408 IC50 = 51 nM T78932 CXJ3I6 117769409 IC50 = 38 nM T78932 C8LTZ6 117769464 IC50 = 29 nM T78932 C4KL1Y 117769470 IC50 = 8.6 nM T78932 CQ46WT 117769476 IC50 = 36 nM T78932 CSKO30 117769533 IC50 = 60 nM T78932 C6XC3W 117769575 IC50 = 7.5 nM T78932 CS95HO 117769592 IC50 = 47 nM T78932 C0PIL5 117769623 IC50 = 34 nM T78932 CO3DA2 117769866 IC50 = 0.92 nM T78932 CI46CP 117770056 IC50 = 1100 nM T78932 C7NI8L 117770083 IC50 = 9.7 nM T78932 CJ3QC8 117770200 IC50 = 770 nM T78932 CSD47C 117770482 IC50 = 1.5 nM T78932 C8SNB9 117770595 IC50 = 9.9 nM T78932 CJ1V9A 117770654 IC50 = 6.7 nM T78932 CS8E6M 117770678 IC50 = 370 nM T78932 CM7X9N 117770754 IC50 = 6.3 nM T78932 C4CFG6 117770831 IC50 = 91 nM T78932 C0X1EQ 117809257 IC50 = 7 nM T78932 CDUH09 117809287 IC50 = 5.7 nM T78932 C45RCJ 118072307 IC50 = 1.6 nM T78932 CH7LT6 118072319 IC50 = 16 nM T78932 CGQK96 118115537 IC50 > 10000 nM T78932 C2OX1Q 118115706 IC50 > 10000 nM T78932 CWCO47 118115913 IC50 > 10000 nM T78932 C72LYV 118116131 IC50 > 10000 nM T78932 C4JW5D 118116385 IC50 > 10000 nM T78932 C34YXR 118139924 Ki = 0.2 nM T78932 C43HNW 118473488 IC50 = 60 nM T78932 CNX7M9 118473558 IC50 = 1.3 nM T78932 CIVS69 118475644 IC50 = 140 nM T78932 CE49ZI 118475652 IC50 = 407 nM T78932 CWQ36P 118475893 IC50 > 3000 nM T78932 CN04RH 118475894 IC50 > 3000 nM T78932 C2P0CG 118475938 IC50 = 3120 nM T78932 CLTV08 118690376 IC50 = 2.1 nM T78932 CRK6J2 118690573 IC50 = 230 nM T78932 CTR74C 118690690 IC50 = 110 nM T78932 CY7BI2 118706214 IC50 > 10000 nM T78932 CI5W9H 118720010 Ki = 16 nM T78932 C5K2QD 118723914 IC50 = 16 nM T78932 C59YJC 118723915 IC50 = 8 nM T78932 C2ON7Y 118723916 IC50 = 680 nM T78932 C5U8WG 118723917 IC50 = 130 nM T78932 C0ZMR8 118723918 IC50 = 210 nM T78932 C4Z5LJ 118723919 IC50 = 280 nM T78932 C85ELI 118723920 IC50 = 90 nM T78932 CGW49X 118723921 IC50 = 150 nM T78932 CXC8K9 118723922 IC50 = 190 nM T78932 CR5JD8 118723923 IC50 = 34 nM T78932 C9W1BU 118723924 IC50 = 390 nM T78932 C8JGN7 118868847 IC50 > 200000 nM T78932 C3DK1Q 118868914 IC50 > 200000 nM T78932 CQ1TL7 118879520 IC50 = 279 nM T78932 C5Z0XH 118911481 IC50 = 250 nM T78932 CT4MJ8 118911570 IC50 = 25 nM T78932 CYTV80 121284861 IC50 = 13 nM T78932 C58NUJ 121284991 IC50 = 390 nM T78932 C3J8CT 121285026 IC50 > 10000 nM T78932 CT9H7V 121285043 IC50 = 5.2 nM T78932 CG9Q1H 121320416 IC50 = 132000 nM T78932 C8NYP1 122189151 IC50 = 10 nM T78932 CFU15S 122191618 IC50 = 70 nM T78932 CE4F3A 122191619 IC50 = 1700 nM T78932 CAC5U1 122191620 IC50 = 290 nM T78932 CRF2K0 122191625 IC50 = 2300 nM T78932 CFKD32 122191637 IC50 = 14300 nM T78932 CPY1K9 122191778 IC50 = 5624 nM T78932 C1H4IX 122192065 IC50 = 6400 nM T78932 C98EJO 122192066 IC50 = 2700 nM T78932 CM1XD7 122192067 IC50 = 3100 nM T78932 C0MLH5 122192068 IC50 = 2500 nM T78932 CC4T6A 122192069 IC50 = 3700 nM T78932 CGO6M7 122192070 IC50 = 3300 nM T78932 CBP34K 122192071 IC50 = 4200 nM T78932 CA2TF6 122192072 IC50 = 7500 nM T78932 CFY30Z 122192073 IC50 = 2500 nM T78932 CJ09XF 122192074 IC50 = 3500 nM T78932 C6LS8X 122192075 IC50 = 2700 nM T78932 C7DJA5 122192076 IC50 = 3200 nM T78932 CAS86F 122192079 IC50 = 5800 nM T78932 CG7TP0 122192080 IC50 = 4300 nM T78932 C5K8UM 122192081 IC50 = 2800 nM T78932 CS4XB9 122199230 IC50 > 200000 nM T78932 CNA45R 122362931 IC50 = 78 nM T78932 C68PHW 122579408 IC50 = 13 nM T78932 C5GR4U 122615173 Ki = 0.015 nM T78932 C7X6ZB 122630882 Ki = 0.018 nM T78932 CX37RN 126715380 IC50 = 2800 nM T78932 CR9C1G 127030133 IC50 = 60 nM T78932 C4JF8H 127040661 IC50 = 1280 nM T78932 C7P5MY 127040994 IC50 = 11400 nM T78932 CB2SE8 127049004 IC50 = 30700 nM T78932 CS6ZO5 127049005 IC50 = 31000 nM T78932 C1PE9L 127050562 IC50 = 4300 nM T78932 CZ5D8C 127050563 IC50 = 42200 nM T78932 CX46RS 127050564 IC50 = 25700 nM T78932 C3LI1J 127050565 IC50 = 5600 nM T78932 CG91WC 127052080 IC50 = 4100 nM T78932 CS4JD0 129626433 IC50 = 7 nM T78932 CZ13WL 130339268 IC50 = 17 nM T78932 CD4NY1 131839645 IC50 = 12 nM T78932 C6OXE3 132134663 IC50 = 10 nM T78932 CUO0C5 132156633 IC50 > 10000 nM T78932 CK4FI7 132277003 IC50 > 10000 nM T78932 C3HC0S 134537158 IC50 = 110 nM T78932 CN75GU 134611727 IC50 = 44 nM T78932 C80PJI 134611728 IC50 = 25 nM T78932 CFM46L 134812674 IC50 = 23 nM T78932 CVF86X 135125189 IC50 = 9 nM T78932 C9MCQ0 135138184 IC50 = 13 nM T78932 CPHG43 135567142 IC50 = 1.5 nM T78932 C2NRS8 135567293 IC50 = 9.1 nM T78932 C4R1FH 135567294 IC50 = 54.5 nM T78932 CA0R9G 135567295 IC50 = 815.9 nM T78932 CRI5F3 135839295 IC50 = 102.1 nM T78932 CH8W7B 135839328 IC50 = 291.2 nM T78932 CJID74 136013449 IC50 = 1200 nM T78932 CHA4N2 136013680 IC50 > 10 nM T78932 C1YUD0 136219394 IC50 > 10 nM T78932 CIU8W3 136254389 IC50 > 10 nM T78932 C1P6ZW 136263939 IC50 = 0.8 nM T78932 C0R2IL 136901416 IC50 = 158.49 nM T78932 CIJ71W 137028350 IC50 = 3200 nM T78932 CS15TL 137028351 IC50 = 3700 nM T78932 CE9V4U 137174991 IC50 = 9 nM T78932 CM64UH 137175110 IC50 = 7 nM T78932 C70DIP 137223928 IC50 = 57.5 nM T78932 C9F3KV 137321155 IC50 = 73.66 nM T78932 CJK67W 137321156 IC50 = 39.43 nM T78932 C3Z4AT 137321159 IC50 > 10000 nM T78932 CMY0V2 137321160 IC50 > 10000 nM T78932 CWM9S4 137349398 IC50 = 179 nM T78932 C9I5TJ 137631461 Ki = 8.8 nM T78932 CAM8K0 137632226 IC50 > 200000 nM T78932 CH9WK1 137632228 IC50 > 5000 nM T78932 C7R2HI 137632648 IC50 > 200000 nM T78932 C2I3PY 137633211 IC50 = 2000 nM T78932 CJN68H 137633647 IC50 > 200000 nM T78932 CF6RH5 137633780 IC50 = 1.7 nM T78932 COE76K 137634328 IC50 = 20.1 nM T78932 C6IU0M 137634461 IC50 = 11 nM T78932 CE4DH3 137635161 IC50 > 200000 nM T78932 C6JVG9 137635398 IC50 = 188 nM T78932 CMV38W 137635509 IC50 > 2000 nM T78932 C0VXM3 137635710 Ki = 0.6 nM T78932 CM73AT 137635759 IC50 > 200000 nM T78932 CH5SI7 137636771 IC50 > 200000 nM T78932 C8I2NQ 137637573 IC50 = 240 nM T78932 C3RF7B 137638414 IC50 > 200000 nM T78932 CE0ZF8 137638897 IC50 = 25.1 nM T78932 C50WHR 137641404 IC50 > 200000 nM T78932 C2VWE5 137642024 IC50 > 200000 nM T78932 CJ6PU9 137642141 IC50 = 958.6 nM T78932 C0RX1Z 137642404 IC50 = 4 nM T78932 CVCM89 137642443 Ki = 3500 nM T78932 C9GDQ6 137642740 IC50 = 8 nM T78932 C94ELU 137643208 IC50 > 2000 nM T78932 CO83EQ 137643608 IC50 = 392.3 nM T78932 CQP79B 137643915 IC50 > 200000 nM T78932 CGHP09 137645020 IC50 = 4.6 nM T78932 CN34SE 137646319 IC50 > 2000 nM T78932 CI8S5A 137646690 IC50 > 200000 nM T78932 CQYM31 137646825 Ki = 20 nM T78932 CGE91V 137646834 IC50 > 200000 nM T78932 CE8SH2 137647292 IC50 > 2000 nM T78932 CUA12V 137647912 Ki = 42 nM T78932 CW6D9H 137648009 IC50 > 200000 nM T78932 C9KW2L 137648948 IC50 > 200000 nM T78932 CHN7A3 137648975 IC50 > 200000 nM T78932 CIB60Q 137649981 IC50 = 12 nM T78932 CF4X3E 137650150 IC50 > 10000 nM T78932 CVHT54 137650515 IC50 > 200000 nM T78932 CJQ72A 137650866 IC50 > 10000 nM T78932 CA9K6R 137650880 IC50 > 200000 nM T78932 COCF21 137651256 IC50 = 0.2 nM T78932 C3Z7LM 137651481 IC50 = 3.9 nM T78932 CQ27PY 137651710 IC50 = 796.2 nM T78932 CYA52Z 137652173 IC50 = 14 nM T78932 C6UEB9 137653042 IC50 > 200000 nM T78932 CK81UT 137654424 IC50 > 2000 nM T78932 CW6SO7 137654686 IC50 > 200000 nM T78932 CCR5B3 137654793 IC50 = 144 nM T78932 CKM89A 137654900 IC50 = 13 nM T78932 C26ONG 137654955 IC50 > 200000 nM T78932 CE9OW2 137655154 Ki = 0.8 nM T78932 CVBS03 137656215 IC50 = 0.5 nM T78932 CYWE21 137656346 IC50 = 22.7 nM T78932 C6V3WR 137656619 IC50 > 200000 nM T78932 CT1EP3 137656679 IC50 = 437.5 nM T78932 C8VC9A 137657080 IC50 = 15.3 nM T78932 C49GYQ 137658008 IC50 > 200000 nM T78932 C59BVH 137658028 IC50 = 1.8 nM T78932 C6UM5X 137658102 Ki = 31 nM T78932 CO6C8I 137658504 IC50 > 200000 nM T78932 CW4CK8 137659037 IC50 = 40 nM T78932 C86KOS 137659382 IC50 > 200000 nM T78932 CR41KW 137660124 IC50 = 0.7 nM T78932 CQ8KF2 137660642 IC50 > 200000 nM T78932 CU48TN 137661036 Ki = 17 nM T78932 COMQ54 137661391 IC50 > 200000 nM T78932 CJ52WM 137661888 IC50 > 200000 nM T78932 CO4DP9 137662248 Ki = 1.2 nM T78932 CU2L5H 138108525 IC50 = 459 nM T78932 C2W0JU 138319690 IC50 > 30000 nM T78932 CXV84M 138377596 IC50 = 49 nM T78932 C8X9DR 138584993 IC50 = 273.4 nM T78932 C9NL1M 138585023 IC50 = 2.24 nM T78932 CHX6N7 138585027 IC50 = 4.35 nM T78932 C3RM2Z 138585033 IC50 = 1.93 nM T78932 CBF8S4 138585069 IC50 = 5730 nM T78932 C4O0GC 138585070 IC50 = 18.42 nM T78932 C7KYU3 138585074 IC50 = 336.3 nM T78932 CE5S4Z 138585101 IC50 = 4766 nM T78932 CM63FA 138585111 IC50 = 32.39 nM T78932 C2U8PZ 138585129 IC50 = 17.4 nM T78932 C0Y2WZ 138585150 IC50 = 427.45 nM T78932 CHMX08 138585151 IC50 = 8.38 nM T78932 CA8N5T 138585156 IC50 = 166.85 nM T78932 CG8TR3 138585164 IC50 = 45.1 nM T78932 C3JR7K 138585184 IC50 = 1163.5 nM T78932 CQI78V 138585192 IC50 = 176.3 nM T78932 C2UCN9 138605457 IC50 > 1000 nM T78932 C3RM1U 138605458 IC50 = 708.65 nM T78932 CD4M3W 138605461 IC50 = 256.5 nM T78932 C4VMQ9 138605557 IC50 = 1502 nM T78932 CCKY16 138756256 IC50 = 180 nM T78932 CQ6R7X 138911330 Ki = 0.07 nM T78932 CI7C4P 140943115 IC50 = 32 nM T78932 C3QHX4 140943118 IC50 = 110 nM T78932 CO41GC 140943126 IC50 = 17 nM T78932 CV0J7Y 140943142 IC50 = 50 nM T78932 CQ3HB0 140943145 IC50 = 4 nM T78932 C7U3KH 140943149 IC50 = 220 nM T78932 CU51PI 141531440 IC50 = 1419.7 nM T78932 C81RPA 141531442 IC50 = 3964.8 nM T78932 CAT46B 141531443 IC50 = 1175.5 nM T78932 CN75MA 141728817 IC50 = 94 nM T78932 C7EL5X 141728840 IC50 = 12 nM T78932 C9H8PX 141728841 IC50 = 67 nM T78932 CC03XH 141728860 IC50 = 60 nM T78932 CECS13 141753441 IC50 > 3000 nM T78932 C2XP8N 145953005 IC50 > 30000 nM T78932 C3L8IE 145958641 IC50 = 419 nM T78932 CO05IK 145959360 IC50 = 74 nM T78932 CFY21D 145961655 IC50 = 14 nM T78932 CI9Z7U 145962747 IC50 = 139 nM T78932 CQ86LZ 145963345 IC50 = 791 nM T78932 C5VWH3 145970734 IC50 = 230 nM T78932 C7K1AJ 145971681 IC50 = 46 nM T78932 C7OD0E 145973587 IC50 = 24000 nM T78932 CHVD06 145979212 IC50 > 10000 nM T78932 C7L1IC 145979240 IC50 > 10000 nM T78932 CAJ37B 145979552 IC50 = 4619 nM T78932 CE31VG 145979714 IC50 = 1839 nM T78932 C7N8DU 145980127 IC50 = 9487 nM T78932 CG3M8I 145980160 IC50 = 66 nM T78932 CM31VB 145980561 EC50 = 3.8 nM T78932 C8AMK1 145980722 IC50 = 2010 nM T78932 C81XFH 145980840 IC50 = 4285 nM T78932 C85XBC 145981348 IC50 = 1816 nM T78932 CD4I2X 145981417 IC50 = 15 nM T78932 CK7E5P 145981833 IC50 = 13 nM T78932 C5VF8P 145983087 IC50 = 1722.2 nM T78932 CS1GK8 145983460 IC50 = 2352.1 nM T78932 CG97VS 145983548 IC50 > 3000 nM T78932 CA20KM 145983867 IC50 = 2117.2 nM T78932 C7THN1 145984160 IC50 = 3144 nM T78932 C30EHD 145984172 IC50 > 10000 nM T78932 C42SJR 145984669 IC50 = 3219.4 nM T78932 C67HUC 145984822 IC50 = 2427.4 nM T78932 CG4U3I 145985120 IC50 = 3296.4 nM T78932 CYP36H 145987360 IC50 = 8 nM T78932 CSN8W5 145987530 IC50 = 8 nM T78932 CW7V1O 145987719 IC50 = 12600 nM T78932 CEA20L 145987749 IC50 = 110 nM T78932 C8NEY2 145987871 IC50 > 9443 nM T78932 C4A2KP 145987909 IC50 = 25 nM T78932 C9ZC0H 145987988 IC50 = 24 nM T78932 C9KJ1A 145988137 IC50 = 239 nM T78932 C9BX4U 145988956 IC50 > 10000 nM T78932 CIVK73 145989244 IC50 > 10000 nM T78932 CC8GZ3 145989610 IC50 = 2890 nM T78932 C5I8SR 145989639 IC50 > 10000 nM T78932 C9CMG6 145989684 Ki = 0.13 nM T78932 CIU9W4 145990027 IC50 > 10000 nM T78932 C3HEC4 145990398 IC50 = 500 nM T78932 C3DWZ0 145990496 IC50 > 10000 nM T78932 CTX1A3 145990814 IC50 = 2971 nM T78932 CL68MB 145990931 IC50 = 6 nM T78932 CNG35K 145991262 IC50 > 10000 nM T78932 C0M6LD 145991292 IC50 > 9817 nM T78932 CKGE38 145991618 IC50 = 2517 nM T78932 CI8R6P 145992803 IC50 > 10000 nM T78932 CZ37YN 145992861 IC50 = 6 nM T78932 CD09RT 145992905 IC50 = 79.4 nM T78932 CG21JZ 145993080 IC50 = 22 nM T78932 CR2F1Y 145993348 IC50 = 3372 nM T78932 C51DMH 145993445 IC50 > 10000 nM T78932 C35PRD 145994244 IC50 = 5 nM T78932 CHQU21 146185142 IC50 = 774 nM T78932 C71KXB 146185156 IC50 = 1453 nM T78932 C9IA1X 146185163 IC50 = 794 nM T78932 CS0OL6 146185170 IC50 = 1298 nM T78932 C1IAH7 146185174 IC50 = 2530 nM T78932 CXQE21 154605321 Ki = 0.34 nM T78932 CQ5BE3 154661514 Ki = 0.26 nM T78932 C5T7UA 154701267 Ki = 0.06 nM T78932 C2FD8V 155510753 Ki = 0.07 nM T78932 C3KE8Z 155510943 Ki = 0.12 nM T78932 C7PLT9 155510967 IC50 = 2690 nM T78932 CZ52CM 155511037 IC50 = 150 nM T78932 CR1SE8 155511850 IC50 = 368 nM T78932 CL2P1A 155512660 Ki = 0.38 nM T78932 C4ZYV6 155513034 Ki = 0.13 nM T78932 C2MD1Q 155513187 IC50 > 10000 nM T78932 C43QZB 155513894 IC50 = 270 nM T78932 C6W0RT 155514076 Ki = 0.035 nM T78932 C83ZSG 155514311 IC50 = 63 nM T78932 C7MJY5 155514805 IC50 = 2000 nM T78932 CP53LB 155515726 IC50 = 280 nM T78932 CP95JN 155516134 Ki = 0.091 nM T78932 C9VK3I 155517004 IC50 = 0.49 nM T78932 C2X8HA 155517088 Ki = 0.8 nM T78932 CZ0RI7 155517469 IC50 = 520 nM T78932 C0E7WS 155518120 IC50 = 48 nM T78932 CDTG10 155518349 IC50 = 5 nM T78932 C0A9LX 155520276 IC50 = 7202 nM T78932 C4YJN9 155520341 IC50 = 23 nM T78932 C0YEX7 155521332 IC50 = 210 nM T78932 C3O1NK 155523586 Ki = 0.48 nM T78932 COKA60 155523996 IC50 = 8 nM T78932 CK14UT 155528172 IC50 = 148 nM T78932 CB26JT 155528364 IC50 = 70 nM T78932 CL47NH 155529550 IC50 = 1300 nM T78932 C7J9MU 155531384 IC50 = 1.6 nM T78932 C5V6PY 155532206 IC50 = 33 nM T78932 C4LE7Q 155532724 IC50 = 180 nM T78932 CR5YW9 155533007 IC50 = 140 nM T78932 CLSV71 155533995 IC50 = 510 nM T78932 CD26VI 155534361 IC50 = 1.8 nM T78932 C2NPE6 155534808 IC50 = 160 nM T78932 C64FIW 155534972 IC50 = 702 nM T78932 CF5JH9 155535582 IC50 > 10000 nM T78932 CHOC87 155535920 IC50 = 58 nM T78932 CE8QW2 155535975 IC50 = 20 nM T78932 C5RC0M 155537160 Ki = 0.14 nM T78932 CF7PQ6 155538533 IC50 = 1.5 nM T78932 C5K0RG 155538766 IC50 = 230 nM T78932 C0D8OL 155540191 IC50 = 251.19 nM T78932 C16MHE 155540242 IC50 = 87 nM T78932 CP2NY0 155540484 IC50 = 158.49 nM T78932 CF8O5T 155540488 IC50 = 19952.62 nM T78932 C51JNT 155540621 IC50 = 398.11 nM T78932 CN1CB2 155540954 Ki = 0.74 nM T78932 CY8F7S 155541097 IC50 = 71 nM T78932 CH6LV1 155541475 IC50 = 251.19 nM T78932 CS58BA 155541478 IC50 = 1564 nM T78932 C1B6EK 155542401 IC50 = 398.11 nM T78932 CH59RW 155542578 IC50 = 16 nM T78932 CKL31P 155542961 IC50 = 1000 nM T78932 C1QRZ2 155543349 IC50 = 28 nM T78932 CRA21U 155543538 IC50 > 3000 nM T78932 C8WJ7H 155544232 IC50 = 870 nM T78932 CP7XE1 155545114 IC50 = 630.96 nM T78932 CFR42U 155545338 IC50 = 6309.57 nM T78932 C5BHW8 155546008 IC50 = 0.32 nM T78932 C5U8HP 155546232 IC50 = 398.11 nM T78932 C2Z3PX 155546437 IC50 = 5200 nM T78932 CSI1U9 155547916 IC50 = 55 nM T78932 C0B3RK 155547921 IC50 = 7943.28 nM T78932 CQB92J 155549032 IC50 = 520 nM T78932 C10OSG 155550219 IC50 = 150 nM T78932 C3DW8J 155550308 IC50 = 501.19 nM T78932 C31QUW 155550462 IC50 = 120 nM T78932 C6UJS7 155550600 IC50 = 330 nM T78932 C0DMP2 155551420 IC50 = 2175 nM T78932 C52UAJ 155551442 IC50 = 2500 nM T78932 CD60UK 155551659 Ki = 0.29 nM T78932 CW1UX0 155552333 IC50 = 630.96 nM T78932 CEA05C 155552433 Ki = 0.33 nM T78932 CPB6M8 155553409 IC50 = 1532 nM T78932 C5HQ7X 155553551 IC50 = 27 nM T78932 C3C2LK 155553968 IC50 = 750 nM T78932 CNTP52 155554413 IC50 = 19 nM T78932 CQ6S8E 155554939 IC50 = 501.19 nM T78932 CP39ZD 155555305 IC50 = 794.33 nM T78932 C9J4HM 155555486 IC50 = 201 nM T78932 CG48UE 155556474 IC50 = 316.23 nM T78932 C8TYG7 155556520 IC50 = 1738 nM T78932 CL82WM 155558175 Ki = 0.15 nM T78932 CHW4O3 155558352 IC50 = 316.23 nM T78932 C7WND0 155558729 IC50 = 76 nM T78932 C2U5ZM 155559343 IC50 = 2511.89 nM T78932 CSF54R 155559609 IC50 = 1740 nM T78932 CANJ25 155559746 IC50 = 2511.89 nM T78932 CK0SC3 155560352 IC50 = 33 nM T78932 CNK81M 155560413 IC50 = 794.33 nM T78932 C54NQC 155561203 IC50 = 53 nM T78932 C5N2SZ 155561228 IC50 = 5.9 nM T78932 CDW8A4 155562327 Ki = 0.29 nM T78932 C4X7ZY 155563244 Ki = 0.024 nM T78932 C68TCL 155563799 IC50 = 2290 nM T78932 CBQN81 155564466 IC50 = 2561 nM T78932 CZ2NK9 155565077 IC50 = 6309.57 nM T78932 C4B3XA 155565275 Ki = 0.22 nM T78932 C4VYW0 155565520 IC50 = 160 nM T78932 CSNF76 155565806 IC50 = 794.33 nM T78932 CE03HW 155566039 IC50 = 0.58 nM T78932 CF1X5I 155566525 IC50 = 32 nM T78932 C0L6UT 155568261 IC50 = 316.23 nM T78932 C8EYW3 155568955 IC50 = 2295 nM T78932 C14DIR 16750188 IC50 = 150 nM T78932 C5UI4F 16750189 IC50 = 120 nM T78932 C6JKT9 16750206 IC50 = 70 nM T78932 CYIU14 16750228 IC50 = 79 nM T78932 CX4I6T 16750253 IC50 = 170 nM T78932 CI79TY 16750254 IC50 = 160 nM T78932 CS6UT4 16750288 IC50 = 190 nM T78932 CI67WG 16750292 IC50 = 57 nM T78932 CIGJ63 16750308 IC50 = 71 nM T78932 CL2SY5 16750330 IC50 = 620 nM T78932 CE5P2I 53363072 IC50 = 140 nM T78932 CTV60O 53363073 IC50 = 160 nM T78932 CD74BW 53363074 IC50 = 110 nM T78932 CU3M8P 53363075 IC50 = 140 nM T78932 C07FTA 53363076 IC50 = 470 nM T78932 C9JX2G 53363150 IC50 = 84 nM T78932 CJ04SF 53363151 IC50 = 180 nM T78932 CO7Z2P 53363152 IC50 = 140 nM T78932 C1T2LY 53363154 IC50 = 80 nM T78932 C9GEA7 53363242 IC50 = 81 nM T78932 CTSP38 53363245 IC50 = 18 nM T78932 CM7BZ3 53363246 IC50 = 140 nM T78932 C0QON7 53363337 IC50 = 36 nM T78932 CU76JB 53363338 IC50 = 180 nM T78932 C2PU3M 53364335 IC50 = 5200 nM T78932 C10FXI 53364337 IC50 = 210 nM T78932 C2U9QE 53364338 IC50 = 170 nM T78932 D00ERW 44444843 Ki > 1936 nM T78932 D00HVA 11624601 Ki > 1900 nM T78932 D06HVH 54613583 IC50 > 10000 nM T78932 D06WGX 9549184 IC50 > 25000 nM T78932 D09HVH 135566652 IC50 > 10 nM T78932 D0H7DQ 6419755 IC50 = 2310 nM T78932 D0IR6U 5494425 IC50 = 1 nM T78932 D0OZ2S 11785878 IC50 = 1200 nM T78932 D0Q3NG 11715520 Ki > 1900 nM T78932 D0R2WK 16038120 IC50 = 2309 nM T78932 D0S7IE 11658882 Ki > 1900 nM T78932 D0V6VQ 53344620 IC50 = 1632.2 nM T62184 D0ED7U 60648 Ki = 16.98 nM T62184 D08ESA 198693 IC50 = 260 nM T62184 D0C9XA 119 IC50 = 3000 nM T62184 CJ9V4G 40598 IC50 > 1000000 nM T62184 CZ6MS1 91274 IC50 = 49 nM T62184 C1W5GH 134985 IC50 = 200 nM T62184 CXSD61 155246 IC50 = 96900 nM T62184 CHV0G9 639062 IC50 > 1000000 nM T62184 C97FYX 702501 IC50 > 300000 nM T62184 C8X9TQ 1069892 Ki > 100000 nM T62184 C1A0UL 1502074 IC50 = 2511.89 nM T62184 C3DR8J 1502075 IC50 = 3162.28 nM T62184 C9EI4M 1530639 IC50 > 1000000 nM T62184 CU23IC 4531494 IC50 = 233000 nM T62184 CG1ZF6 5311322 Ki = 27000 nM T62184 CN2C7Q 6604883 IC50 = 439000 nM T62184 C4A6SU 8181355 IC50 > 500000 nM T62184 CQ64IH 9797818 Ki = 72.44 nM T62184 CRB3U5 9867395 IC50 = 39810.72 nM T62184 C31HNE 9884272 Ki > 100000 nM T62184 CY2IS7 9888224 IC50 = 26000 nM T62184 CI06JL 9982662 IC50 = 10000 nM T62184 CTZ5Q7 9983570 IC50 = 268000 nM T62184 C75BDY 10031163 IC50 = 73000 nM T62184 CZ4PO2 10050339 IC50 = 58000 nM T62184 CZQ52G 10052359 IC50 = 121000 nM T62184 CP2WF1 10072112 IC50 = 133000 nM T62184 CG1A4H 10073933 IC50 = 19000 nM T62184 C57RVK 10075407 IC50 = 78000 nM T62184 C4S1CO 10096504 IC50 = 43000 nM T62184 CQ64PJ 10251287 IC50 = 1400 nM T62184 C0XI3N 10252046 IC50 = 5000 nM T62184 CXJR61 10252950 IC50 = 6900 nM T62184 C0I9UT 10387048 IC50 = 3000 nM T62184 CC8V4E 10412575 IC50 = 142000 nM T62184 CZ8FQ2 10481573 IC50 = 122000 nM T62184 C7KEN9 10938177 IC50 = 309.03 nM T62184 CGMH62 11036614 IC50 = 645.65 nM T62184 C5YIF8 11678946 IC50 = 840 nM T62184 CU40KP 11743493 IC50 = 43000 nM T62184 CH6GX1 13314232 IC50 > 500000 nM T62184 C1D5XO 15124790 IC50 > 1000000 nM T62184 CQ6R8N 15355217 Ki = 41.69 nM T62184 CH9Y5B 17159064 IC50 > 400000 nM T62184 C6VK4E 17173775 IC50 > 1000000 nM T62184 CE92MX 17174058 IC50 > 1000000 nM T62184 C3OQD7 17250318 IC50 > 500000 nM T62184 CME93B 43345728 IC50 > 1000000 nM T62184 CA3WV8 44405923 IC50 = 66300 nM T62184 C3LV6B 44405925 IC50 = 27600 nM T62184 C65RPI 44405927 IC50 = 4340 nM T62184 CMZ4J1 44405929 IC50 > 100000 nM T62184 CN3IE2 44406165 IC50 > 100000 nM T62184 C82BRH 44406167 IC50 = 1240 nM T62184 CV6B3R 44406193 IC50 = 12300 nM T62184 C68YIC 44406195 IC50 > 100000 nM T62184 CUPO14 44406208 IC50 > 100000 nM T62184 CA3PZ2 44406212 IC50 > 100000 nM T62184 C57SOK 44406223 IC50 = 940 nM T62184 C5HGJ6 44406227 IC50 = 650 nM T62184 CGL8E9 44406233 IC50 > 100000 nM T62184 CA5M0R 44406250 IC50 = 2800 nM T62184 CD4O2U 44406255 IC50 = 7100 nM T62184 C3DMC7 44406257 IC50 = 680 nM T62184 C1Y4FA 44406260 IC50 = 1360 nM T62184 CT1P3H 44406279 IC50 = 340 nM T62184 C9W7YV 44406301 IC50 = 1500 nM T62184 C5JUW9 47058964 IC50 > 1000000 nM T62184 CLIK30 50941729 Ki = 14.79 nM T62184 CC5W7V 53317293 Ki = 138.04 nM T62184 C6RXP5 53317294 Ki > 10000 nM T62184 CQMI12 53317407 Ki = 1071.52 nM T62184 CVCF51 53318538 Ki = 61.66 nM T62184 C4MD9S 53318587 Ki = 19.05 nM T62184 C1IPA8 53318588 Ki = 38.9 nM T62184 CF2XU8 53318650 Ki = 371.54 nM T62184 CS2YW1 53318651 Ki = 1905.46 nM T62184 C0RN2B 53318700 Ki = 691.83 nM T62184 C7KX1J 53318701 Ki = 93.33 nM T62184 CH8V2S 53318777 Ki = 93.33 nM T62184 C6O4HV 53319862 Ki = 56.23 nM T62184 C3PS8I 53319863 Ki = 354.81 nM T62184 C7HX1A 53319971 Ki = 102.33 nM T62184 C23CPL 53321157 Ki = 58.88 nM T62184 C2OKR1 53321158 Ki = 46.77 nM T62184 C3LSO8 53321159 Ki = 158.49 nM T62184 C8ST1B 53321160 Ki = 38.02 nM T62184 C4QR9P 53321215 Ki = 18.2 nM T62184 CVPD82 53321216 Ki = 53.7 nM T62184 CPW0R2 53321217 Ki = 831.76 nM T62184 C7TQN0 53321279 Ki = 165.96 nM T62184 CJN7E6 53321326 Ki = 645.65 nM T62184 C19VGM 53321703 Ki = 20.42 nM T62184 CVK6O1 53322546 Ki > 10000 nM T62184 CHN27L 53322918 Ki > 10000 nM T62184 C2O4NS 53323872 Ki > 10000 nM T62184 CL8O7M 53323981 Ki = 69.18 nM T62184 CR68SQ 53325105 Ki = 89.13 nM T62184 CQ03OL 53325106 Ki = 70.79 nM T62184 C5PZR6 53325157 Ki = 52.48 nM T62184 CA0U3E 53325158 Ki > 10000 nM T62184 COXL71 53325159 Ki > 10000 nM T62184 C7S6WZ 53325277 Ki = 28.84 nM T62184 CDP45Q 53325278 Ki = 29.51 nM T62184 CYD14T 53326404 Ki = 331.13 nM T62184 C5ES8V 53326405 Ki = 33.88 nM T62184 C2GYR5 53326406 Ki = 77.62 nM T62184 C63MIE 53326407 Ki = 72.44 nM T62184 CI5BY7 53326408 Ki = 380.19 nM T62184 CDA2N4 53326453 Ki = 2754.23 nM T62184 CG5AL9 53326506 Ki = 199.53 nM T62184 C3G6LJ 53326507 Ki = 676.08 nM T62184 C1WX0P 53326550 Ki = 371.54 nM T62184 CS03PY 53326631 Ki = 40.74 nM T62184 CUB9V6 53326792 Ki = 380.19 nM T62184 C0MRI8 53326796 Ki = 21.88 nM T62184 CQ4XJ7 55285849 IC50 > 100000 nM T62184 CY9O8W 55285850 IC50 > 100000 nM T62184 C8UTR2 67642717 IC50 = 71400 nM T62184 C6ME5H 70684991 IC50 = 809000 nM T62184 C79CYX 70689234 IC50 = 632000 nM T62184 CD9EV5 70691307 IC50 = 270000 nM T62184 CJ7P8C 70691309 IC50 = 270000 nM T62184 C53QGB 118711599 IC50 > 100000 nM T62184 C74FVZ 118727501 Ki = 3981.07 nM T62184 C8I7FR 118727502 Ki = 213.8 nM T62184 CZO19U 118727503 Ki = 1096.48 nM T62184 CT4S7P 118727504 Ki = 66.07 nM T62184 CCR7Q3 118727512 Ki = 20417.38 nM T62184 C9FMU8 118727514 Ki = 19054.61 nM T62184 CO18BS 137635197 IC50 > 1000000 nM T62184 CQL64H 137637846 IC50 > 1000000 nM T62184 CZ73DV 137638595 IC50 > 100000 nM T62184 CARI53 137638617 IC50 > 100000 nM T62184 CUM2T0 137638836 IC50 > 100000 nM T62184 C3PY5G 137638838 IC50 > 50000 nM T62184 CP7OV5 137639241 IC50 > 100000 nM T62184 C21IZT 137639281 IC50 > 1000000 nM T62184 CP24OX 137642163 IC50 > 100000 nM T62184 CK2VU3 137650102 IC50 > 1000000 nM T62184 CJYI80 137650733 IC50 > 1000000 nM T62184 C52PYO 137650910 IC50 > 1000000 nM T62184 CS6FX4 137651374 IC50 > 1000000 nM T62184 CPLJ94 137651669 IC50 > 1000000 nM T62184 CN04QK 137652511 IC50 > 1000000 nM T62184 CGC1Z4 137654858 IC50 > 50000 nM T62184 CADN74 137657292 IC50 > 100000 nM T62184 C4NK1W 137658990 IC50 > 50000 nM T62184 CPI4S8 137659917 IC50 > 50000 nM T62184 CL0U5M 155511885 IC50 = 169824.37 nM T62184 CI7S8H 155516242 IC50 > 100000 nM T62184 C4U8QT 155524561 IC50 > 100000 nM T62184 CJ4OV6 155530359 IC50 > 100000 nM T62184 C4RL9X 155535776 IC50 > 100000 nM T62184 CBR16K 155543188 IC50 = 42657.95 nM T62184 CI30JH 155544639 IC50 = 134896.29 nM T62184 C6OME4 155548176 IC50 = 134896.29 nM T62184 CQD12U 155558328 IC50 = 169824.37 nM T62184 CEP8F2 155559550 IC50 = 134896.29 nM T62184 CL2Q6G 155567178 IC50 > 100000 nM T62184 D02ANG 5216267 IC50 = 158489.32 nM T62184 D03IWW 6575389 IC50 = 116000 nM T62184 D08YGM 92409 IC50 = 130 nM T62184 D0D2EF 1796510 IC50 = 5960 nM T62184 D0H7WK 10458835 IC50 > 100000 nM T62184 D0P3KI 9888030 IC50 = 11400 nM T62184 D0RF2M 4498 IC50 = 8000 nM T62184 D0V5OY 16725912 Ki > 100000 nM T62184 D0V7RG 3532 IC50 = 14000 nM T62184 D0X3CF 442879 IC50 = 20600 nM T45262 D05IIN 5282340 Ki = 2 nM T45262 D07QWW 9888194 Ki = 4 nM T45262 D08UYM 9801039 IC50 = 4 nM T45262 D0LI1C 44469321 IC50 > 30000 nM T45262 D0ZC0M 11596613 Ki = 6.31 nM T45262 D0ZM5O 9884366 IC50 = 4.5 nM T45262 D01KKE 11223423 IC50 = 66.07 nM T45262 D03KJS 177990 Ki = 0.84 nM T45262 D07NWC 9934089 Ki = 3.7 nM T45262 D0G0GI 9909468 Ki = 1.7 nM T45262 D0R2KV 9818802 IC50 = 6.8 nM T45262 C9M4PE 1799074 Ki = 216 nM T45262 C1KW2N 1799083 Ki = 1459 nM T45262 CZ7K9U 3568686 Ki = 2720 nM T45262 C94YQI 3623188 Ki = 2285 nM T45262 CU6X7G 3983703 Ki > 10000 nM T45262 C6UQ2R 4183319 Ki = 15 nM T45262 CL68RO 4596095 Ki > 10000 nM T45262 CM1K7I 9797993 Ki = 57 nM T45262 CM3B8Q 9798798 Ki = 14.5 nM T45262 CJ3RO8 9800789 Ki = 130 nM T45262 CJ4MB8 9801390 Ki = 4.2 nM T45262 C4UC9V 9801874 Ki = 2.3 nM T45262 CI7NP0 9802053 Ki = 2.9 nM T45262 CBX35T 9803011 Ki = 9.4 nM T45262 C8LH0Q 9803645 Ki = 11.2 nM T45262 CK6L2B 9803991 Ki = 68 nM T45262 CH01CO 9805117 Ki = 23.9 nM T45262 CO9VA3 9820671 IC50 = 3.4 nM T45262 CUJ9M1 9821153 Ki = 32 nM T45262 CDM54E 9821250 Ki = 2.6 nM T45262 C2HYB3 9821586 Ki = 0.9 nM T45262 CT8UY2 9822241 Ki = 1 nM T45262 C3ZMR6 9824147 Ki = 8.6 nM T45262 CIZ08K 9824168 Ki = 5.1 nM T45262 C18KSV 9824227 Ki = 1.9 nM T45262 CC93UK 9827578 IC50 = 49 nM T45262 C5V8LW 9828534 Ki = 32 nM T45262 CM64TS 9828535 Ki = 32 nM T45262 CFV16R 9843355 Ki = 3.3 nM T45262 C0J7SB 9843598 Ki = 2 nM T45262 CL0B6C 9843717 Ki = 16.2 nM T45262 CZKS51 9843989 Ki = 158.49 nM T45262 CCTM38 9844591 Ki = 13.1 nM T45262 C2IOY1 9846806 Ki = 13 nM T45262 CQ5F1H 9849255 Ki = 6.6 nM T45262 CQB86U 9865060 IC50 = 50.12 nM T45262 CQI43C 9865133 Ki = 26 nM T45262 CGC08L 9865345 Ki = 62 nM T45262 C07SOD 9865434 Ki = 44 nM T45262 C0U9SC 9865575 Ki = 15 nM T45262 CKJ10P 9865624 Ki = 3.4 nM T45262 C2A5PU 9865886 IC50 = 123.03 nM T45262 CMN1D6 9866114 Ki = 13 nM T45262 C2KV6H 9866408 Ki > 10000 nM T45262 CVP45N 9867507 Ki = 10.5 nM T45262 C9DTJ6 9868427 Ki = 4.1 nM T45262 C10HTZ 9869432 Ki = 8.6 nM T45262 CVO4K6 9870876 Ki = 45.4 nM T45262 CIRH02 9884878 Ki = 1 nM T45262 CDJ7A2 9885480 Ki = 3 nM T45262 CA8CX9 9886113 Ki = 9 nM T45262 CU4S2A 9887145 Ki = 12 nM T45262 CLE15J 9887524 Ki = 63.1 nM T45262 CL78GT 9890659 Ki = 122 nM T45262 CDN73C 9891049 Ki = 8 nM T45262 CTY7S5 9907170 Ki = 12 nM T45262 C1AIV4 9908466 Ki = 4.4 nM T45262 C4R9LK 9908879 Ki = 0.5 nM T45262 C7SMT0 9908904 IC50 = 4.7 nM T45262 C93VNK 9909978 Ki = 0.62 nM T45262 C35KUD 9910700 Ki = 6.1 nM T45262 CEW89P 9912040 Ki = 4.6 nM T45262 CGFU68 9912938 Ki = 3.1 nM T45262 CW5LY9 9913240 Ki = 1.1 nM T45262 CW9RC7 9928790 Ki = 507 nM T45262 C7HR3F 9929418 Ki = 9.2 nM T45262 C6N3LE 9931098 Ki = 4.4 nM T45262 C8PA3R 9931738 Ki = 5 nM T45262 C61JWZ 9931767 Ki = 1.7 nM T45262 CF0P8C 9931814 Ki = 1.9 nM T45262 CUG0B5 9932463 Ki = 7.5 nM T45262 CX9DL7 9933199 Ki = 5.012 nM T45262 C3ES2F 9935525 Ki = 5 nM T45262 C40WKE 9945957 Ki = 23.7 nM T45262 C63ISH 9946605 Ki = 14.4 nM T45262 C98FOI 9950645 Ki = 90 nM T45262 CQZ3H2 9950788 Ki = 2.4 nM T45262 CBT9J8 9951076 Ki = 4.2 nM T45262 C64FSL 9951620 Ki = 60 nM T45262 C8PI2R 9952376 Ki = 3.3 nM T45262 CEF6H1 9952997 Ki = 1.585 nM T45262 C2ESG8 9954503 Ki = 17 nM T45262 CY7T6V 9955329 Ki = 3 nM T45262 CVTB47 9956594 Ki = 4.1 nM T45262 CZP23J 9957261 Ki = 12.6 nM T45262 C1NT0V 9957428 Ki = 14.5 nM T45262 CF2G3N 9957619 Ki = 7.4 nM T45262 CF2EI5 9960282 Ki = 3.2 nM T45262 C2ZK7A 9969024 Ki = 5.9 nM T45262 C14KGN 9970050 IC50 = 35 nM T45262 C0DX5E 9980256 Ki = 2021 nM T45262 C3F7HW 9980267 Ki = 22 nM T45262 C9A5QZ 9980466 Ki = 11 nM T45262 C9HK1C 9998456 Ki = 8000 nM T45262 CLWN39 10024020 Ki = 11 nM T45262 CYBX45 10025032 Ki = 456 nM T45262 COZ8R9 10026532 Ki = 9 nM T45262 CBC2F6 10027220 Ki = 2.4 nM T45262 C0X1GR 10028059 Ki = 2 nM T45262 C1KT6Q 10041172 Ki = 35 nM T45262 CVD19S 10048451 Ki = 30 nM T45262 CI0W2P 10048452 Ki = 22 nM T45262 CZ3CT5 10075105 IC50 = 30 nM T45262 C9FMO5 10095518 Ki = 2.4 nM T45262 C8O6EA 10110271 IC50 = 170 nM T45262 CLA9Y0 10111093 Ki = 0.4 nM T45262 C4NY2A 10111096 Ki = 19.2 nM T45262 CYZ2G0 10111139 EC50 = 80 nM T45262 CPL75J 10112758 IC50 = 490 nM T45262 C2FJB9 10113422 Ki = 6700 nM T45262 CM2N4P 10117501 Ki = 120 nM T45262 CVE87C 10118581 Ki = 6300 nM T45262 CK4M7P 10119101 Ki = 25 nM T45262 C3B8KJ 10132995 Ki = 15 nM T45262 CM1DG3 10133826 Ki = 22 nM T45262 C4RY9N 10135080 IC50 = 38 nM T45262 CPH83V 10135150 IC50 = 22 nM T45262 CERU90 10136000 Ki = 1.6 nM T45262 CWA30V 10138067 Ki = 9 nM T45262 COU34K 10140223 Ki = 1100 nM T45262 CB60DK 10142098 Ki = 6.3 nM T45262 CIF3K0 10142769 Ki = 110 nM T45262 CA1KP5 10155816 Ki = 46 nM T45262 COBC76 10155870 Ki > 10000 nM T45262 CABI02 10157369 Ki = 5000 nM T45262 CW4BK7 10160871 Ki = 11000 nM T45262 CE25KB 10163122 Ki = 26 nM T45262 C8FA0P 10164483 Ki = 290 nM T45262 CJ8M6G 10164617 Ki = 43 nM T45262 CM37OX 10164848 Ki = 56 nM T45262 CG4WX9 10165732 Ki = 37 nM T45262 C0YAV4 10166079 Ki = 390 nM T45262 C8TO0N 10166565 Ki = 50 nM T45262 CRUA85 10177704 IC50 = 37 nM T45262 CQ32YN 10178818 Ki = 5.6 nM T45262 C83JBE 10178898 IC50 = 37 nM T45262 CM47RT 10180350 IC50 = 31.62 nM T45262 CZL36A 10180472 Ki = 2800 nM T45262 C3CB1P 10183075 Ki = 290 nM T45262 C7DUR1 10186078 Ki = 130 nM T45262 CT8R1C 10188470 Ki = 3.7 nM T45262 C7VD6N 10200119 Ki > 5000 nM T45262 CJQ6O1 10200135 IC50 = 15 nM T45262 CLC9J3 10200724 Ki = 4.4 nM T45262 CQ6B8T 10204577 Ki = 1800 nM T45262 C9PRM8 10204603 IC50 = 25.12 nM T45262 CKC48Q 10204820 Ki = 67 nM T45262 C4YDO1 10205521 Ki = 5.7 nM T45262 CX42DA 10206448 Ki = 420 nM T45262 CM78RQ 10206904 Ki = 560 nM T45262 CNSU91 10207702 Ki = 100 nM T45262 CEB6R9 10222402 IC50 = 80 nM T45262 CF9H8L 10222698 Ki = 1150 nM T45262 C0ZT4O 10222795 EC50 = 200 nM T45262 CK27YW 10223332 Ki = 4.1 nM T45262 CVL14I 10224173 Ki = 1.8 nM T45262 C6PZL4 10228046 Ki = 31000 nM T45262 CEBW73 10228129 Ki = 6 nM T45262 CTQ75B 10229290 Ki = 1300 nM T45262 C6VFU4 10255153 IC50 = 23 nM T45262 CUPM27 10268909 Ki = 354 nM T45262 CWU94F 10273816 Ki = 16000 nM T45262 COM25X 10275456 Ki = 150 nM T45262 CBRC42 10276375 Ki = 160 nM T45262 C3I6PU 10277733 IC50 = 15.85 nM T45262 C1QM4S 10277887 Ki = 73 nM T45262 C4HA9Z 10292638 Ki = 2600 nM T45262 C4JZ5H 10294046 IC50 = 600 nM T45262 CT3R6P 10294626 Ki = 0.7 nM T45262 C97MQK 10295219 Ki = 6.1 nM T45262 CZN71G 10295681 Ki = 820 nM T45262 C4B6FR 10297799 Ki = 51000 nM T45262 C05PDF 10298157 Ki = 100 nM T45262 CD5C1O 10298158 Ki = 23 nM T45262 CEG5L7 10299169 Ki = 5100 nM T45262 CID9P2 10300313 Ki = 12 nM T45262 CYQ4P6 10301060 Ki = 38 nM T45262 C8OUJ7 10302495 Ki = 11 nM T45262 C9IX0A 10303191 Ki = 6.1 nM T45262 CMC02R 10303689 Ki = 4.8 nM T45262 CZQ1G2 10316753 Ki = 2400 nM T45262 C5SA0X 10319873 Ki = 35 nM T45262 CUP85M 10366978 Ki = 5 nM T45262 C1IK8Y 10367821 Ki = 5.5 nM T45262 CHW4N6 10388138 Ki = 0.9 nM T45262 CPJ1Z0 10402860 Ki = 43 nM T45262 C0RDL7 10410573 Ki = 53 nM T45262 CAM37Z 10428930 Ki = 1 nM T45262 C65GOT 10474043 Ki = 15 nM T45262 CG1YN0 10477079 Ki = 436 nM T45262 CO1E7F 10479355 Ki = 1.5 nM T45262 CR1FC4 10498852 Ki > 100 nM T45262 CK83AH 10500067 Ki = 7 nM T45262 CPZ5R2 10500190 Ki = 20.7 nM T45262 CF69CA 10500311 Ki = 416 nM T45262 C91QHI 10501205 Ki = 194 nM T45262 CY07OC 10501643 Ki = 24 nM T45262 C20GXT 10502620 Ki = 150 nM T45262 C1W0AK 10502738 Ki = 4 nM T45262 CK38AN 10503074 Ki = 5 nM T45262 C1NM8L 10503714 Ki = 7.1 nM T45262 C7Z1GI 10504356 Ki = 25 nM T45262 C6JZL3 10504455 Ki = 20.4 nM T45262 C4VPE0 10506052 Ki = 14 nM T45262 C6HED9 10526779 Ki = 44 nM T45262 CTF04S 10526864 Ki = 28 nM T45262 CPNG38 10527467 Ki = 5 nM T45262 CNV21E 10527943 Ki = 38.7 nM T45262 CYIB57 10528499 Ki = 235 nM T45262 CXE21P 10528542 Ki = 9.8 nM T45262 CNPS51 10528613 Ki = 66.9 nM T45262 CF1T3Z 10529311 Ki = 14 nM T45262 C85GVL 10542924 Ki = 1050 nM T45262 C42BTC 10546541 Ki > 10000 nM T45262 CVW0E3 10547488 Ki = 490 nM T45262 CJ34IM 10548253 Ki > 10000 nM T45262 C4N7AV 10548395 Ki = 1050 nM T45262 CS1I7H 10548743 Ki = 8 nM T45262 C1M8EA 10549179 Ki = 5.2 nM T45262 CVEK14 10549365 Ki = 6 nM T45262 CN5I7U 10549751 Ki = 46 nM T45262 C5TI4L 10549928 Ki > 1000 nM T45262 COR01G 10549983 Ki = 291 nM T45262 C15ZVH 10549990 Ki = 22 nM T45262 CA87MF 10550438 Ki = 3.8 nM T45262 CIR8J6 10550837 Ki = 3460 nM T45262 CJ7QH6 10551312 Ki = 4.3 nM T45262 C0D6BI 10551475 Ki = 203 nM T45262 C3TF1Y 10552046 Ki = 21.3 nM T45262 CHP81W 10552437 Ki = 4.5 nM T45262 CD47RK 10552595 Ki = 123 nM T45262 CV8N1R 10552787 Ki = 0.8 nM T45262 C4LC3H 10553475 Ki = 41 nM T45262 C8GTF4 10563926 Ki > 1000 nM T45262 C67YER 10565818 Ki > 10000 nM T45262 C2YC5X 10567951 Ki = 115 nM T45262 CZ4WP3 10571912 Ki = 8 nM T45262 CXV78I 10572455 Ki = 33 nM T45262 C7SFD4 10573027 Ki = 30 nM T45262 CNI2B4 10573028 Ki = 70 nM T45262 CV4C2L 10573217 Ki = 25.3 nM T45262 CH3JE1 10574875 Ki = 10.6 nM T45262 C84XIJ 10575478 Ki = 64 nM T45262 CE38FX 10576086 Ki = 10.5 nM T45262 CW8T3L 10576982 Ki = 9 nM T45262 C2F1PV 10593122 Ki = 5.7 nM T45262 CFM31Y 10593782 Ki > 10000 nM T45262 CV73BX 10594766 Ki = 1470 nM T45262 CO2K1V 10595854 Ki = 10 nM T45262 CO38VZ 10596113 Ki = 15 nM T45262 C0EJG3 10596146 Ki = 25 nM T45262 CL13MJ 10598041 Ki = 287 nM T45262 CZD0L3 10599448 Ki = 2665 nM T45262 C4SL9D 10616065 Ki > 10000 nM T45262 CR0L5C 10616216 Ki = 130 nM T45262 C9PGN6 10617667 Ki > 10000 nM T45262 CRBO48 10618927 Ki = 27.3 nM T45262 CVY82F 10621342 Ki = 27 nM T45262 CF9C0D 10622505 Ki = 83 nM T45262 CZEQ68 10622522 Ki = 3.2 nM T45262 C10PCT 10622647 Ki = 8 nM T45262 C98RJW 10623894 Ki = 476 nM T45262 CHUC73 10624822 Ki > 1000 nM T45262 C8T6MF 10638639 Ki > 10000 nM T45262 CCXW41 10641809 Ki > 10000 nM T45262 CQ8HW0 10643831 Ki = 13 nM T45262 CU03ZM 10645784 Ki = 41 nM T45262 C6XA2F 10646276 Ki = 5 nM T45262 C9AGM4 10646364 Ki = 24 nM T45262 C8XZM0 10646423 Ki = 9.7 nM T45262 C08JDK 10646531 Ki = 5 nM T45262 CS7E8M 10646985 Ki = 2.9 nM T45262 CR40VT 10647940 Ki = 17 nM T45262 C3G8ML 10648379 Ki = 31.3 nM T45262 C04LBW 10648981 Ki = 1.4 nM T45262 CJW37B 10662222 Ki = 60 nM T45262 CEBI87 10664736 Ki = 68 nM T45262 CS70LV 10665582 Ki = 29 nM T45262 C0QEM9 10666336 Ki > 100 nM T45262 CYO3J6 10667231 Ki > 100 nM T45262 CAL16S 10667354 Ki = 1.1 nM T45262 CE3S9V 10667355 Ki = 26 nM T45262 COR8M2 10667729 Ki = 24.1 nM T45262 C6FTR2 10668220 Ki = 1.2 nM T45262 C8D2LQ 10668655 Ki = 253 nM T45262 C20KBU 10668656 Ki > 10000 nM T45262 C0O7GK 10669045 Ki = 17 nM T45262 C0E2GX 10669526 Ki = 120 nM T45262 CV15FY 10670904 Ki = 3.9 nM T45262 CN8LR2 10671608 Ki = 32.5 nM T45262 C3KFH7 10671924 Ki = 100 nM T45262 C0I8FP 10672237 Ki = 6.7 nM T45262 CA49UJ 10672294 Ki = 39.7 nM T45262 CH1LP4 10686834 Ki = 90 nM T45262 CK7CV0 10686839 Ki = 36 nM T45262 C96GSN 10688248 Ki = 35 nM T45262 CW0CT7 10690278 Ki = 7.6 nM T45262 C4GVB0 10692645 Ki = 242 nM T45262 C7KY0Q 10692703 Ki = 1.6 nM T45262 C3PBL2 10693263 Ki = 5.2 nM T45262 C6OIT0 10694122 Ki = 5 nM T45262 C03JRW 10694584 Ki = 0.9 nM T45262 CA8EO0 10694630 Ki = 3.1 nM T45262 C5SKU0 10694719 Ki = 19.4 nM T45262 C9NUO6 10695347 Ki = 4.7 nM T45262 CWI36G 10708209 Ki = 54 nM T45262 CV3N1I 10710543 Ki = 20 nM T45262 CMYH95 10712065 Ki = 7.1 nM T45262 CZN65C 10715520 Ki = 0.6 nM T45262 CO24TV 10717499 Ki = 4.4 nM T45262 C4QF6S 10717500 Ki = 4.3 nM T45262 C5MR7X 10717531 Ki = 15.3 nM T45262 C7BL6P 10717634 Ki = 9 nM T45262 CDT9Q4 10717814 Ki = 21 nM T45262 COK4E1 10736859 Ki = 20.7 nM T45262 C4H7YU 10738874 Ki > 10000 nM T45262 CQJ4A1 10739468 Ki = 11 nM T45262 CQ7H0Z 10739593 Ki = 2.2 nM T45262 C69PDR 10739849 Ki = 12.4 nM T45262 CA01KW 10739909 Ki = 69.6 nM T45262 C0VPW4 10740327 Ki = 7.1 nM T45262 C4MKL8 10740981 Ki = 10 nM T45262 CSG74V 10741252 Ki = 4.7 nM T45262 CX0HT7 10741433 Ki = 195 nM T45262 CLNT70 10741479 Ki = 4 nM T45262 C6N3MY 10741540 Ki = 22 nM T45262 CSFE76 10761294 Ki = 201 nM T45262 CE3A5Y 10763375 Ki = 44.5 nM T45262 CR26ZU 10764399 Ki = 27.7 nM T45262 C4Y5PR 10764802 Ki = 6 nM T45262 C5RDC3 10765120 Ki = 33.7 nM T45262 CHOP92 10765122 Ki = 3 nM T45262 C8F7ZD 10766371 Ki = 22 nM T45262 CA1X9R 10782323 Ki > 10000 nM T45262 CJF4C0 10783164 Ki = 5700 nM T45262 CJZS53 10784215 Ki = 27.5 nM T45262 C63ZTA 10785716 Ki = 1700 nM T45262 CPU5F4 10786785 Ki = 1.9 nM T45262 CE6VJ4 10786789 Ki = 51 nM T45262 C8TKE4 10787219 Ki = 1690 nM T45262 CLIF25 10787254 Ki = 2.5 nM T45262 CLUD85 10788201 Ki = 25.3 nM T45262 COVT84 10788803 Ki = 2.8 nM T45262 C4QF9V 10788999 Ki = 6 nM T45262 C7ET5A 10789145 Ki = 6.2 nM T45262 CBR2Z0 10789622 Ki = 3.5 nM T45262 CN9L2O 10789842 Ki = 23.5 nM T45262 CD51ZL 10790231 Ki = 1026 nM T45262 C02JUS 10790606 Ki = 4 nM T45262 CG1X5U 10791657 Ki = 33.2 nM T45262 CDL71Y 10807869 Ki = 25 nM T45262 C91DGW 10807999 Ki > 10000 nM T45262 CFA52M 10808132 Ki = 23 nM T45262 CC12PF 10808133 Ki = 490 nM T45262 C93IMF 10808915 Ki = 4 nM T45262 CWV98K 10809350 Ki > 10000 nM T45262 CGS69N 10809708 Ki = 5 nM T45262 C6RAL8 10810752 Ki = 20 nM T45262 C40SZO 10811877 Ki = 29 nM T45262 CMAV90 10812125 Ki = 15.4 nM T45262 CMAS64 10813254 Ki = 1.5 nM T45262 CQ5YP6 10813394 Ki = 10.3 nM T45262 CD2H4X 10813479 Ki = 26 nM T45262 CPC68Q 10813902 Ki = 5.9 nM T45262 C0W6YE 10828446 Ki > 1000 nM T45262 CYO57R 10828851 Ki > 10000 nM T45262 C8FY1O 10830877 Ki = 1390 nM T45262 CQ1DI7 10831985 Ki = 59.4 nM T45262 CY18RU 10832574 Ki = 1.2 nM T45262 CEI6P5 10832987 Ki = 7 nM T45262 C41ZTP 10833915 Ki = 3918 nM T45262 CB9D5M 10835052 Ki = 2 nM T45262 CPQW50 10835160 Ki = 27 nM T45262 CD51AO 10835652 Ki = 55000 nM T45262 CXV74P 10835759 Ki = 3.5 nM T45262 CP4SG6 10835789 Ki = 3.5 nM T45262 CQXA68 10836468 Ki = 9.2 nM T45262 C5RV7X 10837003 Ki = 5.1 nM T45262 CT7O9J 10838302 Ki = 5 nM T45262 C1OI4H 10838946 Ki = 36.7 nM T45262 C53PBY 10853581 Ki = 1204 nM T45262 C64KLM 10854115 Ki > 10000 nM T45262 C6KW9O 10857993 Ki = 6230 nM T45262 CP2D1L 10870698 Ki > 10000 nM T45262 C24VLI 10892583 Ki = 2261 nM T45262 CPRM34 10902707 Ki = 115 nM T45262 C2ZPF3 10904621 Ki > 10000 nM T45262 C1SI7V 10913225 Ki > 10000 nM T45262 C6JR4L 10914632 Ki = 291 nM T45262 CEC39W 10926611 Ki > 10000 nM T45262 C6E9IH 10946918 Ki = 415 nM T45262 CU0IG5 10948253 Ki > 10000 nM T45262 CU7G3V 10957905 Ki > 10000 nM T45262 C7G6ZW 10958631 Ki > 10000 nM T45262 CSCN68 10958953 Ki = 8600 nM T45262 CQ87NV 10969620 Ki > 10000 nM T45262 C0MAN7 10969667 Ki > 10000 nM T45262 C7ZA9G 10969669 Ki > 10000 nM T45262 C9ABT8 10970599 Ki > 10000 nM T45262 CL7TH6 10981146 Ki > 10000 nM T45262 CU94DT 10991736 Ki = 6953 nM T45262 CPU5Q3 11001793 Ki > 10000 nM T45262 C42PUT 11012118 Ki > 10000 nM T45262 CCB1U2 11022343 Ki = 526 nM T45262 CA2KV4 11022531 Ki = 299 nM T45262 C5LPO4 11023489 Ki > 10000 nM T45262 CG1ER4 11032842 Ki = 4708 nM T45262 CZ6R1H 11034476 Ki = 652 nM T45262 C18IEA 11045497 Ki = 417 nM T45262 CBC4L3 11046479 Ki = 538 nM T45262 CKS16N 11046519 Ki > 10000 nM T45262 CFP91Y 11055441 Ki > 10000 nM T45262 C3LRU7 11065415 Ki = 526 nM T45262 C4KLW3 11065773 Ki = 1079 nM T45262 CFN6R1 11067569 Ki = 51 nM T45262 CIW69A 11077161 Ki = 62 nM T45262 CIPG26 11078292 Ki = 197 nM T45262 C8C0VO 11087955 Ki > 10000 nM T45262 CX65WP 11089973 Ki > 10000 nM T45262 C7A2QZ 11101179 Ki > 10000 nM T45262 CYBR08 11109264 Ki = 1403 nM T45262 C4WZX3 11119591 Ki > 10000 nM T45262 C4AZ7H 11120236 Ki > 10000 nM T45262 C9U5XB 11120577 Ki > 10000 nM T45262 C8W6AE 11121533 Ki > 10000 nM T45262 CM98ZX 11122528 Ki = 38 nM T45262 C7Z9AU 11141163 Ki = 1832 nM T45262 CM0DR9 11152649 Ki = 30 nM T45262 CJ1P4B 11153216 Ki = 20 nM T45262 CVO6S4 11153312 EC50 = 0.7 nM T45262 CUD32C 11153953 Ki = 40 nM T45262 CX6FQ5 11154954 Ki = 460 nM T45262 CIW7B2 11155555 Ki = 428 nM T45262 C6CF0T 11156095 Ki = 55 nM T45262 C46BAS 11164902 Ki = 10 nM T45262 C91JZR 11165678 Ki = 5.7 nM T45262 CD98BW 11166658 Ki = 13 nM T45262 C3GL9U 11166919 Ki = 6 nM T45262 C0G9BU 11175998 Ki = 49 nM T45262 C7XY4R 11177298 Ki = 4.2 nM T45262 C10JSF 11178281 Ki = 22 nM T45262 C6N9UZ 11178740 Ki = 4 nM T45262 CAU90J 11182525 Ki > 1000 nM T45262 C3D2RZ 11188091 Ki = 190 nM T45262 CV1O4G 11188634 Ki = 60 nM T45262 CA8O7M 11189570 Ki = 11 nM T45262 C5YR3P 11189666 Ki = 3.5 nM T45262 CM9OV5 11189676 IC50 = 1230.27 nM T45262 CHE9Z0 11200917 IC50 = 794.33 nM T45262 CA48GU 11201203 Ki = 5.2 nM T45262 C50SEK 11201828 IC50 = 32.36 nM T45262 C7F4QB 11210737 IC50 = 15 nM T45262 CE0HS9 11211248 Ki = 260 nM T45262 C97UNC 11212115 Ki = 14 nM T45262 CT4P2D 11221437 Ki > 10000 nM T45262 C45ZTK 11222685 Ki = 62 nM T45262 C1QS5G 11222924 Ki = 200 nM T45262 CW8Y9Q 11223591 Ki = 1900 nM T45262 C4L5QS 11223627 Ki = 120 nM T45262 CQL43N 11224120 Ki = 2.4 nM T45262 CBI6D2 11224781 Ki = 4.2 nM T45262 CF7MV4 11228715 Ki = 36.7 nM T45262 C2VON4 11235359 Ki = 8.8 nM T45262 CZI4Q9 11235365 Ki = 39 nM T45262 CRV1H0 11235455 IC50 = 316.23 nM T45262 CM29HP 11235868 Ki = 16 nM T45262 CU2DT6 11236249 Ki = 1.3 nM T45262 C2UI0B 11236939 Ki = 16.3 nM T45262 CGJH23 11245503 Ki = 1.7 nM T45262 CJC7I2 11246476 Ki = 1000 nM T45262 CXV9P0 11246568 Ki = 23 nM T45262 C97KWN 11247120 Ki = 32.5 nM T45262 CZM94G 11247393 Ki = 2.3 nM T45262 CUX3C1 11247672 IC50 = 309.03 nM T45262 CC4SE1 11247792 Ki = 46 nM T45262 C7B9CN 11257259 Ki = 4100 nM T45262 CULO20 11268730 Ki = 58 nM T45262 CU7T6E 11271502 IC50 = 65 nM T45262 CYB8N4 11274927 Ki > 1000 nM T45262 CT57VZ 11280879 Ki = 13 nM T45262 CS70DR 11282181 Ki = 2.9 nM T45262 CS34XL 11282792 IC50 = 120.23 nM T45262 C7SM5V 11282946 Ki = 24 nM T45262 CG58CW 11291132 Ki = 85 nM T45262 C9Q5MG 11291949 Ki = 2.2 nM T45262 CPX1O2 11297873 Ki > 1000 nM T45262 C9F0HL 11303504 Ki > 10000 nM T45262 CON72R 11304752 Ki = 920 nM T45262 C0BO5J 11305029 Ki = 3.4 nM T45262 C35QSH 11305354 Ki = 7.3 nM T45262 CD0E8Z 11306179 Ki = 2.7 nM T45262 CE6OG0 11306515 Ki = 13 nM T45262 C8CRJ1 11317069 IC50 = 67.61 nM T45262 CBZL20 11320856 Ki = 45.1 nM T45262 CAC94F 11326060 Ki = 9.4 nM T45262 C7ERU5 11326483 Ki = 20 nM T45262 CV2PK7 11326815 Ki = 2.6 nM T45262 C7U9TK 11328374 Ki = 6.3 nM T45262 CCLW63 11338351 Ki = 9 nM T45262 C1P7SO 11338604 IC50 = 120.23 nM T45262 CKTD58 11339333 Ki = 6.8 nM T45262 COYB67 11348744 Ki = 8800 nM T45262 CDS85I 11350066 Ki = 26 nM T45262 C2E6FO 11350078 IC50 = 67.61 nM T45262 CM9G7S 11351594 Ki = 24 nM T45262 CXKM07 11355390 Ki > 1000 nM T45262 CR96GQ 11361057 Ki = 150 nM T45262 CO8C4W 11362799 Ki = 5.4 nM T45262 CQ9W4F 11372928 Ki = 5.6 nM T45262 C6S2UY 11374063 IC50 = 56.23 nM T45262 CB65JM 11375016 Ki = 15 nM T45262 C9YIW1 11383383 Ki = 46 nM T45262 CRAV61 11383650 EC50 = 4 nM T45262 C01FOV 11383809 Ki = 80 nM T45262 C9CYR1 11383860 Ki = 5.2 nM T45262 C19UWI 11384238 Ki = 3.4 nM T45262 CX6KC0 11386550 Ki = 5.2 nM T45262 CIV8E9 11393576 Ki = 21 nM T45262 CGU83H 11394728 Ki = 26 nM T45262 CUI3Z1 11395654 Ki = 350 nM T45262 C68GLZ 11417694 Ki = 4 nM T45262 C5A3FN 11427630 Ki = 2600 nM T45262 CH5IF6 11429073 Ki = 150 nM T45262 CH4JB2 11429341 Ki = 4.8 nM T45262 C4UC8J 11429605 Ki = 170 nM T45262 CAK84C 11430299 Ki = 2.4 nM T45262 CGS60H 11431638 Ki = 11.7 nM T45262 CY5L3V 11438679 Ki > 10000 nM T45262 CHNC92 11440355 Ki = 910 nM T45262 CW6LD2 11441103 IC50 = 1949.84 nM T45262 CT5C2M 11441193 Ki = 120 nM T45262 C3QGK2 11441545 Ki = 190 nM T45262 C93EYI 11442212 Ki = 14 nM T45262 CI7FY5 11450550 Ki = 690 nM T45262 CFZ5N2 11450996 Ki = 7.3 nM T45262 CT74ZG 11453549 Ki = 84 nM T45262 C7TPX5 11462455 Ki = 1.6 nM T45262 C1A2XQ 11465828 Ki = 2.5 nM T45262 C2QZN8 11474047 Ki = 8 nM T45262 C1ML3I 11474841 Ki = 51 nM T45262 C9R0GA 11475328 Ki = 140 nM T45262 C9FP8B 11475476 IC50 = 50.12 nM T45262 CXC69B 11476167 IC50 = 3235.94 nM T45262 CKV67C 11477320 Ki = 6.5 nM T45262 CANG56 11485413 Ki = 17 nM T45262 CV7Q3I 11486120 Ki = 440 nM T45262 CRQ4B3 11491865 Ki > 1000 nM T45262 CWCL92 11501973 Ki = 31.62 nM T45262 CVPI27 11502109 Ki = 42 nM T45262 CE5Y3L 11509641 Ki = 31.62 nM T45262 CU3N8A 11509708 Ki = 10 nM T45262 CT7FB8 11509709 Ki = 100 nM T45262 CNV2K7 11516283 Ki = 79.43 nM T45262 C20ZEV 11524791 Ki = 7.943 nM T45262 CVFJ80 11524923 Ki = 158.49 nM T45262 CCFD79 11525846 Ki = 7.943 nM T45262 CN9K0P 11530590 Ki = 12.59 nM T45262 C6DJ8W 11531570 Ki = 31.62 nM T45262 CL0RW9 11531898 Ki = 50.12 nM T45262 CJ8SY4 11538121 Ki = 63.1 nM T45262 CT2CG1 11545949 Ki = 7.943 nM T45262 C4S2FU 11546255 Ki = 0.2 nM T45262 C2BXA9 11552261 EC50 = 4.1 nM T45262 C97QFN 11560105 Ki = 7.943 nM T45262 CVT4I2 11560698 Ki = 3.981 nM T45262 C5L4ZF 11568262 Ki = 19.95 nM T45262 CB6L0C 11575986 Ki = 10 nM T45262 C0ON7E 11576870 Ki = 6.31 nM T45262 C1OK6W 11588927 IC50 = 2.4 nM T45262 C72YMN 11589539 Ki = 5.012 nM T45262 C6YJ1G 11598576 Ki = 3.981 nM T45262 C0HE9D 11598824 Ki = 50.12 nM T45262 C54DYC 11602680 Ki = 794.33 nM T45262 C6WI7Q 11605928 Ki = 3.981 nM T45262 CFP23O 11610200 Ki = 5011.87 nM T45262 C3IXU5 11625175 Ki = 12.59 nM T45262 CM56BD 11628147 Ki = 3.981 nM T45262 CR90DB 11634953 Ki = 6.31 nM T45262 CS53HB 11639435 Ki = 10 nM T45262 CO8U1N 11639510 IC50 = 120 nM T45262 CH8KN6 11639847 Ki = 25.12 nM T45262 C2X0AC 11653680 Ki = 63.1 nM T45262 C6WUP7 11656502 Ki = 15.85 nM T45262 CC9D3N 11660986 Ki = 50.12 nM T45262 CGU07M 11677548 Ki = 398.11 nM T45262 CPF9R7 11684703 Ki = 125.89 nM T45262 CZB7H3 11689443 Ki = 94 nM T45262 CV84BR 11691278 Ki = 7.943 nM T45262 CO25PQ 11697131 Ki = 251.19 nM T45262 CPJ21B 11703243 Ki = 79.43 nM T45262 C5NW9X 11703582 EC50 = 5.6 nM T45262 CJQC07 11704536 Ki = 158.49 nM T45262 CGZ45A 11706059 Ki = 79.43 nM T45262 CRVW63 11710664 Ki = 7.943 nM T45262 C61XSQ 11713007 Ki = 3.162 nM T45262 CXL7W6 11713460 Ki = 19.95 nM T45262 CR8S2P 11718607 Ki = 5.012 nM T45262 CY4WX6 11727011 Ki = 3867 nM T45262 CB0ZN5 11728273 Ki > 10000 nM T45262 C05RYO 11742775 Ki = 509 nM T45262 CX23ZM 11749772 Ki = 40 nM T45262 C50SGM 11751039 IC50 = 371.54 nM T45262 C04EIW 11751120 Ki = 7.2 nM T45262 C4G8JM 11751505 Ki = 240 nM T45262 C3PRT0 11759092 Ki = 5 nM T45262 C8FTX2 11759733 Ki = 66 nM T45262 CK42EQ 11773421 Ki = 2.6 nM T45262 CI4O0R 11773483 Ki = 9.1 nM T45262 CGJ4Z2 11774042 Ki = 1.3 nM T45262 COA3Y0 11778680 Ki = 43 nM T45262 C51GBE 11781604 Ki > 10000 nM T45262 CEQ26N 11782614 Ki = 1422 nM T45262 C1SE8P 11782743 Ki > 10000 nM T45262 CGV59J 11792386 Ki = 65 nM T45262 CYJ76C 11792683 Ki = 31 nM T45262 CKGR60 11794714 Ki > 10000 nM T45262 CG45CD 11795486 Ki = 210 nM T45262 CNP07F 11795557 Ki = 5 nM T45262 CYH92P 11795560 Ki = 22 nM T45262 CKV54Q 11796523 Ki = 48 nM T45262 C75QGP 11796930 Ki = 5 nM T45262 CNL09V 11797409 Ki = 24 nM T45262 CFR94O 11797750 Ki = 11 nM T45262 C18CXP 11797773 Ki = 23.8 nM T45262 CB0K2M 11798114 Ki = 6.1 nM T45262 CG0PA1 11798634 Ki = 31 nM T45262 CVXT23 11798911 Ki = 133 nM T45262 CZ5J3M 11798947 Ki = 28.3 nM T45262 CDK37E 11823320 Ki > 10000 nM T45262 CL3UX5 11823600 Ki > 10000 nM T45262 C6WLE3 11948286 IC50 = 4.1 nM T45262 CFG9C3 11983528 IC50 = 144.54 nM T45262 CYJ7B1 12086065 Ki = 5.1 nM T45262 CB01YW 12967647 Ki = 360 nM T45262 CL5F9I 12967650 Ki = 23 nM T45262 CSY24U 12967651 Ki = 100 nM T45262 CS1MO5 12967652 Ki = 79 nM T45262 C0YWC4 12967653 Ki = 28 nM T45262 CS1Y4N 12982784 Ki = 69 nM T45262 CN94EU 15486940 Ki = 1.5 nM T45262 CT2Q4B 15490815 Ki = 24 nM T45262 CR74MI 15490817 Ki = 8.6 nM T45262 C7V6UI 15490818 Ki = 9.1 nM T45262 CT67RZ 15490819 Ki = 369 nM T45262 CLXY34 15490820 Ki = 4.6 nM T45262 C4B3SL 15490822 Ki = 2.5 nM T45262 C3CK5I 15490823 Ki = 20.6 nM T45262 CL0P5E 15965420 Ki = 23 nM T45262 CEC0Y6 16126888 EC50 = 4.9 nM T45262 C1MB4F 16416344 Ki = 310 nM T45262 CY23WI 16730517 Ki = 7.8 nM T45262 CBL8O9 17961227 IC50 = 100 nM T45262 C03QYC 18449319 Ki = 7.3 nM T45262 CBYD90 18449326 Ki = 224 nM T45262 CK34UX 18449330 Ki = 3.7 nM T45262 C42ZPD 18629227 Ki = 1.3 nM T45262 CTQX61 18672241 Ki = 57 nM T45262 CGY4U7 18672249 Ki = 130 nM T45262 C8KQ4U 18672262 Ki = 240 nM T45262 C9DYR1 18672270 Ki = 770 nM T45262 CZA50D 18672272 Ki = 46 nM T45262 CWK1D9 18691298 Ki = 9.7 nM T45262 C1BXW4 18691301 Ki = 95.5 nM T45262 C0MOH7 18691303 Ki = 23.1 nM T45262 CO9V1J 18691306 Ki = 11.2 nM T45262 CK7M0B 18691308 Ki = 60.3 nM T45262 C8TXV1 18691310 Ki = 202 nM T45262 C6LQM1 18691311 Ki = 54.8 nM T45262 CR1V2I 18691315 Ki = 3536 nM T45262 C1JM6Z 18691318 Ki = 18.4 nM T45262 CGS9V3 18691320 Ki = 5.8 nM T45262 CP25GS 18691321 Ki = 78.2 nM T45262 C5O8XN 18691322 Ki = 168 nM T45262 CG7KA1 18691324 Ki = 5.8 nM T45262 CPMH27 18691325 Ki = 9.4 nM T45262 CJD74Q 18691327 Ki = 23.4 nM T45262 C38LKM 18691329 Ki = 32.3 nM T45262 C3H0QF 18691332 Ki = 2359 nM T45262 CO2JE7 19063905 Ki = 49 nM T45262 CHB29S 20779996 Ki = 180 nM T45262 CDG20F 20780008 Ki = 61 nM T45262 CZ8NE3 20780009 Ki = 33 nM T45262 CDVS72 20780016 Ki = 26 nM T45262 C5AW6C 20780017 Ki = 126 nM T45262 C95WFG 20780021 Ki = 270 nM T45262 C0FHQ2 20780024 Ki = 1559 nM T45262 C7TXQ9 20780026 Ki = 41 nM T45262 C5TW2G 20780028 Ki = 94 nM T45262 CE69LG 20780033 Ki = 4200 nM T45262 CNH81J 20780034 Ki = 100 nM T45262 C1IMO8 20780036 Ki = 220 nM T45262 CG6WP5 20780037 Ki = 61 nM T45262 CB5CJ0 20780038 Ki = 220 nM T45262 C0V9SA 20780039 Ki = 1700 nM T45262 CA85JN 20780041 Ki = 240 nM T45262 C4L5PU 20780048 Ki = 8.4 nM T45262 C39DFW 20780049 Ki = 580 nM T45262 C5QW8D 20780050 Ki = 700 nM T45262 CJI30H 20780051 Ki = 48 nM T45262 C7O3HK 20780052 Ki = 700 nM T45262 C80ADE 20780053 Ki = 1300 nM T45262 CE90IP 20780054 Ki = 1400 nM T45262 C4U0KD 20780055 Ki = 2700 nM T45262 C1UON3 20780056 Ki = 1200 nM T45262 C9Q7MS 20780057 Ki = 2800 nM T45262 C1VA6T 20780058 Ki = 570 nM T45262 CI0HF9 20780059 Ki = 3200 nM T45262 C8P4WT 20780060 Ki = 28 nM T45262 CG6R2C 20780061 Ki = 4100 nM T45262 CXW4F6 20780064 Ki = 11 nM T45262 CXHP98 20780065 Ki = 34 nM T45262 CMI13G 20780066 Ki = 7.1 nM T45262 CPZ82Q 20780067 Ki = 53 nM T45262 C3W9ZP 20780068 Ki = 457 nM T45262 CK91OA 20780069 Ki = 653 nM T45262 COX43Q 20780070 Ki = 618 nM T45262 C2YG9P 20780071 Ki = 744 nM T45262 CT9S4X 20780072 Ki = 573 nM T45262 CGVB61 20780073 Ki = 138 nM T45262 CT9SG4 20780074 Ki = 13 nM T45262 CZ60CH 20780075 Ki = 428 nM T45262 C6FZ0M 20780080 Ki = 23 nM T45262 CTD3X8 20780089 Ki = 26 nM T45262 CEB97K 20780105 Ki = 54 nM T45262 C38FKU 20780117 Ki = 7708 nM T45262 CE2LS9 20780120 Ki = 704 nM T45262 CRGP75 20780122 Ki = 36 nM T45262 CU5SK0 20780123 Ki = 18 nM T45262 CH3BK4 20780124 Ki = 360 nM T45262 C8ED9A 20780125 Ki = 570 nM T45262 C9CML2 20780126 Ki = 3560 nM T45262 CBD7L6 20780127 Ki = 1180 nM T45262 C93VZW 20780131 Ki = 4049 nM T45262 CRF4W6 20780133 Ki = 28 nM T45262 CZA3M2 20780137 Ki = 26 nM T45262 CY53UO 20780138 Ki = 75 nM T45262 CX21IO 20780139 Ki = 75 nM T45262 C4BGX6 20780140 Ki = 370 nM T45262 CI1W9L 20780142 Ki = 15 nM T45262 C7JA1G 20780144 Ki = 17 nM T45262 CK9ZN0 20780148 Ki = 11 nM T45262 CV3N8O 20780149 Ki = 362 nM T45262 C2EH1U 20780150 Ki = 43 nM T45262 C8PJ1X 20780153 Ki = 15 nM T45262 CLOR59 20780154 Ki = 410 nM T45262 C1DX3O 20780155 Ki = 250 nM T45262 C2NFC4 20780156 Ki = 1600 nM T45262 C3CAO2 20780161 Ki = 41 nM T45262 CS8Z5I 20780164 Ki = 11 nM T45262 CKZV09 20780165 Ki = 15 nM T45262 C9HIC3 20780167 Ki = 68 nM T45262 C52UIC 20780170 Ki = 2774 nM T45262 CQ7S9B 20780173 Ki = 28 nM T45262 CPE5R1 20780175 Ki = 93 nM T45262 C29OGS 20780177 Ki = 36 nM T45262 COL6C1 20780178 Ki = 20 nM T45262 CTNV34 20780180 Ki = 1412 nM T45262 C2GYJ7 20780182 Ki = 50 nM T45262 CJZ9L8 20780184 Ki = 249 nM T45262 C8F9KD 20780186 Ki = 360 nM T45262 C8NO9Q 20780249 Ki = 650 nM T45262 C2DXL1 20780250 Ki = 770 nM T45262 C78WRX 20780251 Ki = 610 nM T45262 CW7R4C 20780253 Ki = 16 nM T45262 CU48RZ 20780254 Ki = 5.3 nM T45262 CRC5G9 20780255 Ki = 9.1 nM T45262 CM3U4S 20780256 Ki = 270 nM T45262 CNFQ78 20780257 Ki = 3000 nM T45262 CZ81DR 20780265 Ki = 34 nM T45262 CHO65I 20780266 Ki = 13 nM T45262 C57AOS 20780267 Ki = 5.2 nM T45262 CQP84Y 20780269 Ki = 740 nM T45262 C2Q0WE 20780271 Ki = 660 nM T45262 CK9J5G 20780272 Ki = 4100 nM T45262 CZ9SU6 20780274 Ki = 290 nM T45262 CGSR49 20780276 Ki = 24 nM T45262 CT1FV2 20780278 Ki = 75 nM T45262 C6LF4A 20780279 Ki = 41 nM T45262 C98KBX 20780280 Ki = 63 nM T45262 C5ZG7W 20780281 Ki = 73 nM T45262 CSA18I 20780282 Ki = 220 nM T45262 C20MNA 20780283 Ki = 2300 nM T45262 CW9P0S 20780284 Ki = 19000 nM T45262 CMBD32 20780285 Ki = 6600 nM T45262 CFU7Q0 20780286 Ki = 1200 nM T45262 C5JGE6 20780287 Ki = 68 nM T45262 CH79NX 20780288 Ki = 3400 nM T45262 C24NOM 20780290 Ki = 3000 nM T45262 CT8PS1 21084107 IC50 = 200 nM T45262 CGFW45 21916073 Ki = 67 nM T45262 CD1Y4F 21916075 Ki = 245 nM T45262 C6KY7Q 21916077 Ki = 920 nM T45262 CTH19R 21916078 Ki = 31 nM T45262 C3VIZ8 21916094 Ki = 49 nM T45262 C5C8WU 21916104 Ki = 310 nM T45262 CG3OK6 21916107 Ki = 13 nM T45262 C1CO0B 21916109 Ki = 150 nM T45262 CBSX05 21916111 Ki = 69 nM T45262 C0BF2J 21916125 Ki = 260 nM T45262 CH0BL2 21916134 Ki = 13 nM T45262 CTMZ47 21916145 Ki = 32 nM T45262 C6YIF7 21916146 Ki = 53 nM T45262 CDAQ91 21916154 Ki = 59 nM T45262 C5YAZ9 21916155 Ki = 441 nM T45262 CY3G9H 21916156 Ki = 350 nM T45262 CL1VH2 21916165 Ki = 150 nM T45262 CLS0Q3 21916183 Ki = 63 nM T45262 CD3Y4N 21916208 Ki = 21 nM T45262 CNS7Y5 21916214 Ki = 38 nM T45262 CMTE57 21916231 Ki = 350 nM T45262 C0P4OY 21916237 Ki = 5600 nM T45262 C4G2YE 21916240 Ki = 4.5 nM T45262 CQBR16 21916241 Ki = 32 nM T45262 CWSD34 21916243 Ki = 350 nM T45262 CJZI45 21916254 Ki = 12 nM T45262 CZUI29 21916258 Ki = 28 nM T45262 CDL93J 21916260 Ki = 21 nM T45262 CWN65I 21916261 Ki = 364 nM T45262 CDM8E0 21916263 Ki = 48 nM T45262 CYC32B 21916268 Ki = 67 nM T45262 C5M1UJ 21916270 Ki = 8.3 nM T45262 CGX60C 21916273 Ki = 580 nM T45262 CMX76B 21916279 Ki = 20 nM T45262 CRS28U 21916286 Ki = 170 nM T45262 C06XEV 21916288 Ki = 160 nM T45262 CO52XV 21916289 Ki = 150 nM T45262 CB6PY5 21916292 Ki = 14 nM T45262 CF13DP 21916296 Ki = 6.4 nM T45262 CQ53SK 21916299 Ki = 160 nM T45262 C31WZP 21916302 Ki = 21 nM T45262 CYZI02 21916306 Ki = 27 nM T45262 C4ONC8 21916308 Ki = 5.9 nM T45262 CMS18O 21916309 Ki = 440 nM T45262 C38AUM 21916311 Ki = 190 nM T45262 C6M7TI 21916321 Ki = 78 nM T45262 CLWJ04 21916322 Ki = 8.2 nM T45262 CV8L1F 21916323 Ki = 610 nM T45262 CK9RQ4 21916331 Ki = 6 nM T45262 CU0EI2 21916338 Ki = 43 nM T45262 C9O0UJ 21916339 Ki = 760 nM T45262 CRDQ40 21916340 Ki = 130 nM T45262 CJAK30 21916343 Ki = 16 nM T45262 C1Y0TP 21984555 IC50 = 41 nM T45262 C8CNK5 21984580 IC50 = 34 nM T45262 CE07ON 21984613 IC50 = 16 nM T45262 CT1HI0 21984648 IC50 = 12 nM T45262 CP4Z0E 21984697 IC50 = 20 nM T45262 C6U2EY 21984718 IC50 = 13 nM T45262 CWO47R 21984746 IC50 = 480 nM T45262 C29GIC 21984762 IC50 = 10 nM T45262 C6TEL4 21984771 IC50 = 24 nM T45262 CNH3V5 21984783 IC50 = 38 nM T45262 CD6KV4 22004628 Ki = 9 nM T45262 C03ZHW 22177742 IC50 = 22 nM T45262 CCR9X4 22177744 IC50 = 15 nM T45262 CIWJ57 22177795 IC50 = 820 nM T45262 C3XQ2M 22177839 EC50 = 640 nM T45262 CUV08F 22177860 IC50 = 59 nM T45262 C0CXU8 22177864 IC50 = 49 nM T45262 CF06PA 22177924 IC50 = 72 nM T45262 CWJ28I 22177936 IC50 = 620 nM T45262 CAQR89 22177988 IC50 = 240 nM T45262 CKG58W 22178019 IC50 = 71 nM T45262 CO06NR 22178115 IC50 = 97 nM T45262 CLX6E7 22248884 Ki = 4.4 nM T45262 C9ZR0H 22248932 Ki = 12 nM T45262 CD0AX3 22248935 Ki = 1.4 nM T45262 C86UHT 22248956 Ki = 151 nM T45262 CR2E8L 22248970 Ki = 401 nM T45262 CC5K0M 22249005 Ki = 167 nM T45262 CS7YE9 22249007 Ki = 54 nM T45262 CH8O5A 22249028 Ki = 7.8 nM T45262 CX5CM2 22249041 Ki = 11.6 nM T45262 CZ9YH8 22249051 Ki = 8.4 nM T45262 CTL04K 22249054 Ki = 2.2 nM T45262 C6SKG3 22249061 Ki = 17.2 nM T45262 C02ZRM 22249074 Ki = 545 nM T45262 CO95AM 22249081 Ki = 1538 nM T45262 CKA53V 22249094 Ki = 4.1 nM T45262 CXN1Y2 22249115 Ki = 71 nM T45262 C6PST0 22249116 Ki = 4.3 nM T45262 COW6A0 22249128 Ki = 2.5 nM T45262 CU3E4M 22249149 Ki = 5.9 nM T45262 CRD0V1 22249156 Ki = 8.6 nM T45262 C1QRJ6 22324320 Ki = 15 nM T45262 C21AYW 22324325 Ki = 310 nM T45262 C5EIV3 22324329 Ki = 38 nM T45262 C39TXW 22324332 Ki = 530 nM T45262 CF54AU 22324333 Ki = 470 nM T45262 C3SB9J 22324337 Ki = 720 nM T45262 CCKV15 22324340 Ki = 72 nM T45262 C7GAN3 22617869 Ki > 10000 nM T45262 CQ1MS6 23000016 Ki = 460 nM T45262 CPD0B1 23068426 Ki = 8 nM T45262 C5CH8E 23567868 IC50 = 93 nM T45262 CX9OY3 23595014 Ki = 4.6 nM T45262 C0I3PU 23595022 Ki = 1.1 nM T45262 CU03HV 23595043 Ki = 1.9 nM T45262 CKDM63 23595046 Ki = 1.3 nM T45262 CE38BG 24180501 IC50 = 3.981 nM T45262 CX7K8I 24758071 EC50 = 3.3 nM T45262 C3QS8R 24758072 EC50 = 1.8 nM T45262 CG1H7M 24758073 EC50 = 6.9 nM T45262 C7M4PU 24758074 EC50 = 2.5 nM T45262 C5RMW3 24758075 EC50 = 11.5 nM T45262 C5ON6Q 24758076 EC50 = 1.9 nM T45262 CBC2Z3 24805438 IC50 = 3400 nM T45262 C1YRC3 24964079 IC50 = 8.6 nM T45262 CD5J1F 24964084 IC50 = 22 nM T45262 C3B1WD 24971237 IC50 = 7 nM T45262 C2N4TA 25114821 EC50 = 3.2 nM T45262 C8CQ4E 25115057 EC50 = 1 nM T45262 C1P3HD 25149257 IC50 = 2754.23 nM T45262 C0K2XY 25149344 IC50 > 10000 nM T45262 C96SXK 25149345 IC50 > 10000 nM T45262 C8CK7P 25150449 IC50 = 426.58 nM T45262 C2K1DB 25150450 IC50 = 8317.64 nM T45262 CV08HY 25150537 IC50 > 10000 nM T45262 CPZI91 25150538 IC50 > 10000 nM T45262 CXIK35 42618174 Ki = 2 nM T45262 CAM63X 42618195 IC50 = 15.2 nM T45262 C8K4UF 42618197 IC50 = 1.2 nM T45262 C7VX9R 44129684 IC50 = 210 nM T45262 CB0C8T 44156254 IC50 = 48 nM T45262 C63RWQ 44194975 IC50 = 4.9 nM T45262 CG2V5U 44194976 IC50 = 1.9 nM T45262 C9C3VZ 44237814 IC50 = 52 nM T45262 C3ND4M 44266401 Ki = 662 nM T45262 C2IHK3 44266431 Ki = 8.4 nM T45262 CY7O8L 44266437 Ki = 17.4 nM T45262 C69PNB 44266439 Ki = 24.9 nM T45262 CH87OP 44266453 Ki = 229 nM T45262 C43XBO 44266463 Ki = 13.5 nM T45262 CJ3M7P 44266473 Ki = 109 nM T45262 CX34VQ 44266481 Ki = 13.9 nM T45262 CR18FP 44266482 Ki = 10.1 nM T45262 CWLM67 44266488 Ki = 21.4 nM T45262 CP93NU 44266496 Ki = 7.8 nM T45262 CWEH39 44266513 Ki = 84.6 nM T45262 C9IGR7 44266524 Ki = 222 nM T45262 CH4F5M 44266555 Ki = 33.4 nM T45262 CBK34Q 44266581 Ki = 2 nM T45262 CKC0D9 44266918 Ki = 81 nM T45262 CC6O9N 44266947 Ki = 5.5 nM T45262 C8ZB4N 44267063 Ki = 3.1 nM T45262 CDNA37 44267064 Ki = 3 nM T45262 CZ1YE8 44267068 Ki = 70.9 nM T45262 C4MV2L 44290322 Ki = 1.1 nM T45262 C3VP8X 44290482 Ki = 2 nM T45262 CR59IB 44290640 Ki = 13.7 nM T45262 C4FH0Y 44305179 Ki = 511 nM T45262 CNDW60 44305202 Ki = 77 nM T45262 CFB7N2 44305208 Ki = 15 nM T45262 CM4V0Z 44305209 Ki = 93 nM T45262 C65ECG 44305246 Ki = 41 nM T45262 CU6EN4 44305255 Ki = 6.4 nM T45262 CNC98M 44305256 Ki = 40 nM T45262 CYH98A 44305523 Ki = 11 nM T45262 C1N5FS 44305524 Ki = 216 nM T45262 C0C9IP 44305545 Ki = 69 nM T45262 C8EK3I 44305971 Ki = 100 nM T45262 CU0D7C 44305973 Ki = 240 nM T45262 CT8QW6 44305974 Ki = 2000 nM T45262 C9G1OQ 44305986 Ki = 250 nM T45262 CSX1Z0 44306162 Ki = 63 nM T45262 CBVW53 44306185 Ki = 460 nM T45262 CRG1S3 44306205 Ki = 860 nM T45262 CL6PI2 44306220 Ki = 19 nM T45262 CUNY38 44306462 Ki = 63 nM T45262 CKC7J4 44306488 Ki = 15 nM T45262 CGR93X 44306534 Ki = 2200 nM T45262 CB4N9Y 44306535 Ki = 700 nM T45262 CP3HZ7 44307474 Ki = 3 nM T45262 CTJZ81 44307478 Ki = 3 nM T45262 CQ79SM 44307479 Ki = 174 nM T45262 CR12NW 44307491 Ki = 2 nM T45262 CIOC16 44307652 Ki = 112 nM T45262 CH03GM 44307653 Ki = 25 nM T45262 C8NHQ1 44307654 Ki = 16 nM T45262 C5M1JW 44307655 Ki = 62 nM T45262 CZ7SV5 44307724 Ki = 4 nM T45262 CMD53Z 44307737 Ki = 10 nM T45262 C12GHS 44307738 Ki = 2 nM T45262 C5UH1E 44307747 Ki = 20 nM T45262 C7MD5T 44307772 Ki = 2207 nM T45262 C5VAN0 44307783 Ki = 7771 nM T45262 CUX2E1 44307784 Ki = 650 nM T45262 CHEC01 44307806 Ki = 11 nM T45262 C6MGH4 44307825 Ki > 5000 nM T45262 CCH47L 44307838 Ki > 5000 nM T45262 C0K5DW 44307854 Ki > 5000 nM T45262 CBVR64 44307855 Ki = 765 nM T45262 C45FGT 44307856 Ki > 5000 nM T45262 C6ZC0M 44307870 Ki = 16 nM T45262 CE61QC 44307879 Ki = 24 nM T45262 C6N2SO 44307892 Ki = 3 nM T45262 C12MRG 44307893 Ki = 192 nM T45262 CE0T7W 44308017 Ki = 15 nM T45262 CU8IH5 44308134 Ki = 561 nM T45262 CH6L2F 44308155 Ki = 115 nM T45262 C4IE6S 44308156 Ki = 145 nM T45262 C4RE5Z 44308157 Ki = 29 nM T45262 CY8AQ0 44308172 Ki = 38 nM T45262 C46LZU 44308187 Ki = 17 nM T45262 CE53VJ 44315264 Ki = 2100 nM T45262 C7R2KB 44315525 Ki = 8000 nM T45262 CY1JI3 44317641 Ki > 10000 nM T45262 CRE9C1 44317643 Ki > 10000 nM T45262 CSGE91 44317646 Ki > 10000 nM T45262 CBX6Y4 44317647 Ki > 10000 nM T45262 CR75GX 44317664 Ki > 10000 nM T45262 CX7Y6H 44317667 Ki = 3295 nM T45262 CB8AS5 44317728 Ki = 469 nM T45262 CPI94C 44317759 Ki = 752 nM T45262 CUK06F 44317760 Ki = 922 nM T45262 CE1V5B 44317800 Ki = 439 nM T45262 C5J3ZV 44317927 Ki > 10000 nM T45262 CH7E1Z 44317955 Ki = 1075 nM T45262 C9AL6T 44317956 Ki > 10000 nM T45262 CCZ46I 44317957 Ki > 10000 nM T45262 C6J3HE 44317962 Ki = 204 nM T45262 C05ERN 44317964 Ki = 7334 nM T45262 C6JRC8 44317974 Ki > 10000 nM T45262 CB3NF1 44317975 Ki > 10000 nM T45262 C4J2VO 44317976 Ki = 387 nM T45262 CW9L1E 44317977 Ki = 641 nM T45262 C4OJ8S 44317983 Ki > 10000 nM T45262 CA07QO 44317986 Ki > 10000 nM T45262 C5ABV7 44318003 Ki > 10000 nM T45262 CH9BP4 44318055 Ki > 10000 nM T45262 CG8OJ1 44318056 Ki = 3346 nM T45262 CYZ2L3 44318064 Ki > 5000 nM T45262 CU3OH1 44318102 Ki = 260 nM T45262 CV3KL8 44318106 Ki = 4 nM T45262 CJK87B 44318109 Ki = 47 nM T45262 C0KC8T 44318119 Ki = 135 nM T45262 CJU3N9 44318122 Ki = 21 nM T45262 CGTW56 44318123 Ki = 4000 nM T45262 CAG83R 44318168 Ki = 39 nM T45262 C8TQ1J 44321641 EC50 = 0.22 nM T45262 C2NHP7 44337106 Ki = 14 nM T45262 C4OPZ3 44337293 Ki = 33 nM T45262 CFAI49 44337304 Ki = 15 nM T45262 CO7Y9B 44337305 Ki = 22 nM T45262 CZE7K8 44337446 Ki = 1500 nM T45262 CKH42A 44337472 Ki = 310 nM T45262 CR8UM5 44337493 Ki = 72 nM T45262 CC4RK3 44337502 Ki = 2200 nM T45262 CP0T9U 44337516 Ki = 3200 nM T45262 CGS3Y8 44337527 Ki = 10 nM T45262 CFA2W8 44337532 Ki > 10000 nM T45262 CA20RD 44337533 Ki = 2600 nM T45262 C0WU4S 44337549 Ki = 120 nM T45262 C6J4YZ 44337577 Ki = 3400 nM T45262 CYVR10 44341452 Ki = 16.1 nM T45262 CH40JI 44341455 Ki = 230 nM T45262 CAC86V 44341456 Ki = 80 nM T45262 CMDL08 44341463 Ki = 81.5 nM T45262 C8WZY4 44341476 Ki = 27.5 nM T45262 CAY58N 44341491 Ki = 4.1 nM T45262 CY3N2H 44341581 Ki = 2.1 nM T45262 C3WDN1 44341612 Ki = 180 nM T45262 CBH75T 44341634 Ki = 140 nM T45262 CTA51R 44341635 Ki = 16 nM T45262 C9MG0X 44341636 Ki = 5.7 nM T45262 C1UCM3 44341663 Ki = 12.1 nM T45262 CSV8B9 44341664 Ki = 3.8 nM T45262 CD2YE4 44341680 Ki = 7 nM T45262 C0PIF4 44341687 Ki = 14.5 nM T45262 C8Z6LE 44341697 Ki = 35 nM T45262 C83UCV 44341712 Ki = 11 nM T45262 CJG69O 44341714 Ki = 9 nM T45262 CWM72B 44341718 Ki = 37 nM T45262 CY7BL3 44341723 Ki = 1.3 nM T45262 C8AVR4 44341728 Ki = 32 nM T45262 C83XOM 44341729 Ki = 32.8 nM T45262 CBR5K9 44341733 Ki = 8.9 nM T45262 C2ZU4Y 44341734 Ki = 64 nM T45262 CO39ED 44341735 Ki = 1.5 nM T45262 C0SFT6 44341736 Ki = 24 nM T45262 CAGL91 44341737 Ki = 4.4 nM T45262 CLY7W8 44341738 Ki = 32.5 nM T45262 CP37UI 44341739 Ki = 4.4 nM T45262 CP70ON 44341743 Ki = 5.7 nM T45262 CE5N3W 44341754 Ki = 3.2 nM T45262 CZ7YU2 44341755 Ki = 59 nM T45262 CDM0C1 44341762 Ki = 12.5 nM T45262 C3NL9S 44341763 Ki = 32 nM T45262 CAB1N9 44341765 Ki = 3 nM T45262 CB8FK1 44341777 Ki = 46 nM T45262 C4OQ3I 44341805 Ki = 9.7 nM T45262 C8J4WM 44341809 Ki = 70 nM T45262 CH54NV 44341813 Ki = 3.7 nM T45262 CVF1J3 44341814 Ki = 8.2 nM T45262 CY96BO 44341815 Ki = 4 nM T45262 C5V3MT 44341816 Ki = 6.7 nM T45262 C1D2AW 44341817 Ki = 10.5 nM T45262 C4IUH6 44341818 Ki = 10.4 nM T45262 C8WM7O 44341823 Ki = 18 nM T45262 C5SAH6 44341832 Ki = 2 nM T45262 CIDM50 44341835 Ki = 9.8 nM T45262 CQ76JT 44341845 Ki = 1.4 nM T45262 C3K6PU 44341855 Ki = 34 nM T45262 CX4M1Y 44341857 Ki = 380 nM T45262 CC4F5Z 44341858 Ki = 11.2 nM T45262 CTK59I 44341861 Ki = 340 nM T45262 C4ZJC1 44341862 Ki = 5.1 nM T45262 CG7SD1 44341874 Ki = 2.5 nM T45262 CZ03VM 44341875 Ki = 4.5 nM T45262 C9ZYN6 44341877 Ki = 2.1 nM T45262 CQ4FU3 44341879 Ki = 2.8 nM T45262 C89CDP 44341892 Ki = 1.2 nM T45262 C3FS5T 44341901 Ki = 4.8 nM T45262 C87OHJ 44341902 Ki = 52 nM T45262 CZ8R6V 44341921 Ki = 1 nM T45262 CR7K1G 44341936 Ki = 1.3 nM T45262 C1K3DN 44341949 Ki = 420 nM T45262 CS2ND4 44341983 Ki = 170 nM T45262 C2FI6W 44342014 Ki = 3.2 nM T45262 C8AU7C 44342015 Ki = 13 nM T45262 CUN87R 44342074 Ki = 2.2 nM T45262 C24EWL 44342075 Ki = 3 nM T45262 C8C4WF 44342084 Ki = 6.5 nM T45262 CGSK71 44347046 Ki = 2.6 nM T45262 CG03OH 44347061 Ki > 10000 nM T45262 C25KEL 44347076 Ki > 10000 nM T45262 C2LH6G 44347078 Ki > 10000 nM T45262 CH5V3M 44347079 Ki > 10000 nM T45262 CM95GI 44347108 Ki = 100 nM T45262 C0WL6S 44347117 Ki = 150 nM T45262 C17YJC 44347137 Ki = 2.4 nM T45262 CLI49Q 44347138 Ki = 1.9 nM T45262 CUN67V 44347139 Ki = 3.9 nM T45262 C94LKM 44347190 Ki = 29 nM T45262 C5IRZ1 44347200 Ki = 1.3 nM T45262 CRTD78 44347202 Ki = 2.4 nM T45262 C17JCP 44347217 Ki = 3.6 nM T45262 C6JB4Y 44347223 Ki = 24 nM T45262 CH6PY1 44347236 Ki = 3.5 nM T45262 C9IBN1 44347356 Ki = 11 nM T45262 CK3Q8I 44347358 Ki > 10000 nM T45262 CG4C8U 44347359 Ki > 10000 nM T45262 C1QIU0 44347388 Ki = 0.73 nM T45262 CH5G7C 44347421 Ki = 43 nM T45262 CV71LW 44347436 Ki = 8.6 nM T45262 CNE5W3 44352349 Ki > 40000 nM T45262 C13DLN 44352358 Ki = 5100 nM T45262 C39IYK 44352370 Ki = 3500 nM T45262 C90HUB 44352382 Ki = 21 nM T45262 CW31DB 44352386 Ki = 16 nM T45262 CZ4QF6 44352436 Ki = 4600 nM T45262 C83WBE 44352437 Ki = 2900 nM T45262 CHQJ78 44352447 Ki = 7.8 nM T45262 CU93PG 44352448 Ki = 60 nM T45262 C30RMY 44352454 Ki = 73 nM T45262 CJ85KR 44352464 Ki = 28 nM T45262 CYN2Z6 44352478 Ki = 28 nM T45262 CIH40A 44379386 Ki = 18 nM T45262 CP5S8L 44379486 Ki = 18 nM T45262 C1IWZ8 44381175 Ki = 48.5 nM T45262 CK7TB0 44381252 Ki = 48.2 nM T45262 CHN28R 44381468 Ki = 8 nM T45262 C9P7HV 44381516 Ki = 3.6 nM T45262 C4R2YL 44384750 Ki = 17.4 nM T45262 C2M1XD 44384779 Ki = 12.2 nM T45262 CWA21C 44384780 Ki = 47.9 nM T45262 CG5HC9 44384801 Ki = 6.1 nM T45262 CSDX38 44384802 Ki = 4.4 nM T45262 C9Z8QP 44384828 Ki = 130 nM T45262 CTS15K 44384893 Ki = 124 nM T45262 CTY6O8 44385463 Ki = 1179 nM T45262 CI6F0Q 44385503 Ki = 42.8 nM T45262 CLQC92 44385520 Ki = 26.2 nM T45262 CLS58V 44385524 Ki = 890 nM T45262 CR35ZE 44385525 Ki = 113 nM T45262 C5DS8V 44385545 Ki = 117 nM T45262 CMW50Y 44385629 Ki = 698 nM T45262 C1NTG6 44386313 Ki = 345 nM T45262 CMC0V8 44386320 Ki = 1.5 nM T45262 CA0UQ2 44386385 Ki = 259 nM T45262 CENM98 44386432 Ki = 3 nM T45262 CV4XP3 44386496 Ki = 31.1 nM T45262 C1DG2B 44387042 Ki = 7.6 nM T45262 C8YXB3 44387103 Ki = 15.1 nM T45262 C2QIF8 44387214 Ki = 463 nM T45262 C4SN6G 44388393 Ki = 61 nM T45262 CDQN34 44388401 Ki = 280 nM T45262 C17CKW 44388403 Ki = 6.9 nM T45262 C5CQ3X 44388407 Ki = 12 nM T45262 C9HG4L 44389050 Ki = 1100 nM T45262 C0XRS7 44389071 Ki = 18000 nM T45262 C6QNG4 44389082 Ki = 13000 nM T45262 C9AO6B 44389083 Ki = 29000 nM T45262 CAXZ14 44389084 Ki = 55000 nM T45262 C3T2JH 44389087 Ki > 10000 nM T45262 CEJH54 44389088 Ki = 9800 nM T45262 C1N9WK 44389097 Ki = 12000 nM T45262 CLW2M7 44389111 Ki = 42 nM T45262 CDZ0N2 44389113 Ki = 19000 nM T45262 C2TVH4 44389125 Ki = 10000 nM T45262 C7UFO2 44390909 Ki > 10000 nM T45262 CJ7N4G 44391045 Ki > 10000 nM T45262 C52VMW 44391046 Ki > 10000 nM T45262 CBHQ75 44391073 Ki > 10000 nM T45262 CU6NQ9 44391086 Ki > 10000 nM T45262 CJIH26 44391118 Ki > 10000 nM T45262 CF37AS 44391122 Ki > 10000 nM T45262 C1YN9J 44392643 Ki = 6.7 nM T45262 C16DOE 44392644 Ki = 19 nM T45262 C24DOB 44392653 Ki = 1.7 nM T45262 CTUL32 44392657 Ki = 14 nM T45262 C94VMI 44392663 Ki = 1.1 nM T45262 C9D5AZ 44392678 Ki = 40 nM T45262 C40RSG 44392681 Ki = 220 nM T45262 C6QZI1 44392687 Ki = 12 nM T45262 CDXN51 44392688 Ki = 3.2 nM T45262 C78KJZ 44392691 Ki = 55 nM T45262 C6R0NX 44392693 Ki = 13 nM T45262 C4UCS2 44392695 Ki = 1.2 nM T45262 CT13HN 44392702 Ki = 3.9 nM T45262 C2NLD7 44392707 Ki = 3.2 nM T45262 CGZ8D6 44392709 Ki = 17 nM T45262 CQ3OA0 44392710 Ki = 100 nM T45262 CUE2X0 44392711 Ki = 0.8 nM T45262 C12OCL 44392722 Ki = 1.2 nM T45262 C1KX4T 44392723 Ki = 78 nM T45262 CVXR85 44392724 Ki = 88 nM T45262 C9HP0M 44392731 Ki = 1200 nM T45262 CF3BZ8 44392734 Ki = 810 nM T45262 C8H7LM 44392736 Ki > 10000 nM T45262 C9D1JG 44392739 Ki = 530 nM T45262 C1GUK4 44392740 Ki = 110 nM T45262 CZ5V1H 44392741 Ki = 10 nM T45262 CL3F9P 44392742 Ki = 90 nM T45262 CH2F0W 44392743 Ki > 10000 nM T45262 CF04JL 44392747 Ki = 380 nM T45262 C6L5JT 44392748 Ki > 10000 nM T45262 C8C0DK 44392749 Ki = 40 nM T45262 CCNY31 44392750 Ki = 1900 nM T45262 C5Y9EK 44392751 Ki = 560 nM T45262 C0KRS4 44392753 Ki = 13 nM T45262 CDWE17 44392758 Ki = 630 nM T45262 CG25TE 44392759 Ki = 5100 nM T45262 C9W2IM 44392760 Ki = 31 nM T45262 CKTV39 44392761 Ki = 26 nM T45262 CFPE81 44392764 Ki = 58 nM T45262 CS17BR 44392766 Ki = 23 nM T45262 CMD01L 44392767 Ki = 25 nM T45262 C2W1MX 44392771 Ki = 1100 nM T45262 CPGQ73 44392772 Ki = 200 nM T45262 C04WHG 44392773 Ki = 38 nM T45262 C8P9HA 44392775 Ki = 480 nM T45262 CQ9HP5 44392776 Ki = 470 nM T45262 C2RKW7 44392777 Ki = 1900 nM T45262 CZEI78 44392781 Ki = 6.2 nM T45262 CCX69B 44392782 Ki > 10000 nM T45262 CKVN69 44392786 Ki > 10000 nM T45262 CS94MP 44392787 Ki = 810 nM T45262 CG9C2T 44392788 Ki = 180 nM T45262 CGN06S 44392800 Ki = 540 nM T45262 C6ONJ1 44392801 Ki = 79 nM T45262 CQR69T 44392802 Ki = 360 nM T45262 C8SF4K 44392804 Ki > 10000 nM T45262 C7TU8P 44392805 Ki = 6.6 nM T45262 CSR24V 44396572 Ki = 6.5 nM T45262 CU2OD0 44397564 Ki = 291 nM T45262 C1RX7G 44397565 Ki = 333 nM T45262 C4E0TV 44397631 Ki = 930 nM T45262 C6OGH2 44397642 Ki = 150 nM T45262 CV8Y2U 44441101 Ki > 10000 nM T45262 CD61GS 44441102 Ki = 2900 nM T45262 C04JOU 44443567 Ki = 401 nM T45262 CT6JC3 44443568 Ki > 10000 nM T45262 CH7Y4M 44443569 Ki > 10000 nM T45262 CW8A7L 44443570 Ki = 711 nM T45262 C4RF3N 44443571 Ki = 1185 nM T45262 C5VIN2 44443572 Ki = 1207 nM T45262 C40RAM 44443574 Ki = 115 nM T45262 C7DCO3 44443575 Ki = 1540 nM T45262 CG57MV 44443577 Ki = 2703 nM T45262 C8FKD6 44443578 Ki = 3382 nM T45262 CE8OV5 44443580 Ki = 3980 nM T45262 CT6U8B 44443581 Ki > 10000 nM T45262 CIPC96 44443582 Ki > 10000 nM T45262 CW1C5B 44443583 Ki > 10000 nM T45262 C7LXY8 44443584 Ki > 10000 nM T45262 CK91AU 44443586 Ki > 10000 nM T45262 CBQ5K6 44443588 Ki > 10000 nM T45262 CX2TZ7 44443589 Ki > 10000 nM T45262 CF0Y5P 44443590 Ki > 10000 nM T45262 CB1R2D 44443591 Ki = 59 nM T45262 CVE0Q4 44443592 Ki = 251 nM T45262 C83BVQ 44443593 Ki = 384 nM T45262 C6D1RC 44443595 Ki = 530 nM T45262 C61OZT 44443597 Ki = 2123 nM T45262 CN2HQ5 44443599 Ki = 2376 nM T45262 CKBQ96 44443602 Ki = 2434 nM T45262 C51DOR 44443605 Ki = 4688 nM T45262 CM7V8A 44443609 Ki = 337 nM T45262 CQ2F3P 44443611 Ki > 10000 nM T45262 CZH12L 44443613 Ki > 10000 nM T45262 CUF1J3 44443615 Ki > 10000 nM T45262 CR83NX 44443618 Ki > 10000 nM T45262 CTA2V3 44443627 Ki = 266 nM T45262 C3ITF2 44443629 Ki > 10000 nM T45262 C2J1ZH 44443630 Ki = 5473 nM T45262 CU3D5W 44443631 Ki > 10000 nM T45262 CNFD25 44443632 Ki = 222 nM T45262 C71AIS 44443634 Ki = 1261 nM T45262 CH1XW6 44443636 Ki = 1217 nM T45262 CUX3Y9 44443637 Ki > 10000 nM T45262 CR59UP 44443640 Ki > 10000 nM T45262 C8CQ0R 44443642 Ki = 472 nM T45262 CMK7R8 44443643 Ki = 67 nM T45262 C2ZR3C 44443644 Ki > 10000 nM T45262 C2AO5M 44443645 Ki = 82 nM T45262 C0XK1I 44443649 Ki = 214 nM T45262 CX89VP 44443650 Ki = 58 nM T45262 C7UF9P 44443654 Ki = 51 nM T45262 C5HSJ9 44443655 Ki > 10000 nM T45262 CQ10ND 44443658 Ki = 1733 nM T45262 C7UEH4 44443661 Ki = 1208 nM T45262 C5XJ2U 44443662 Ki > 10000 nM T45262 C9L3DO 44444312 IC50 = 125.89 nM T45262 CI1N0Z 44444314 IC50 = 39.81 nM T45262 C8T5NP 44444316 IC50 = 12.59 nM T45262 C4N0TK 44444317 IC50 = 12.59 nM T45262 C8LZ1V 44444318 IC50 = 50.12 nM T45262 CV32WU 44444325 IC50 = 79.43 nM T45262 CT5R8W 44444331 IC50 = 125.89 nM T45262 CYK75C 44444335 IC50 = 63.1 nM T45262 C9Y8TL 44444336 IC50 = 39.81 nM T45262 C8M1IP 44444337 IC50 = 158.49 nM T45262 CQWT29 44446715 Ki = 103 nM T45262 CWX32T 44446716 Ki > 10000 nM T45262 CI23VO 44446717 Ki = 1685 nM T45262 CV7GE4 44446718 Ki > 10000 nM T45262 C92XTL 44446719 Ki = 962 nM T45262 CUO5Y9 44446720 Ki = 21 nM T45262 CA2E7Y 44446721 Ki = 28 nM T45262 CP0AS6 44446722 Ki = 36 nM T45262 CV6MB7 44446723 Ki = 42 nM T45262 C4YV8I 44446724 Ki = 17 nM T45262 C8OC9T 44446725 Ki = 6 nM T45262 C1U7WZ 44446726 Ki = 8 nM T45262 CI2V9P 44446727 Ki = 26 nM T45262 C63JFH 44446728 Ki = 49 nM T45262 C0WZ7O 44446729 Ki = 9 nM T45262 C0G9XM 44446730 Ki = 5 nM T45262 C9VZJ0 44446731 Ki = 7 nM T45262 CN1WO2 44446732 Ki = 165 nM T45262 CW0V3S 44446733 Ki > 10000 nM T45262 C2L3RQ 44446734 Ki = 215 nM T45262 CL9HF2 44446735 Ki = 1063 nM T45262 CB2F5Z 44446736 Ki = 265 nM T45262 CCF7Q0 44446737 Ki = 173 nM T45262 CZT1B0 44446738 Ki = 120 nM T45262 CB63AV 44446739 Ki = 524 nM T45262 CG82QL 44446740 Ki = 30 nM T45262 CDC2A5 44446741 Ki = 41 nM T45262 C2G1TC 44446742 Ki = 32 nM T45262 CIS65K 44460195 Ki > 10000 nM T45262 C5KS3D 44460259 Ki = 3180 nM T45262 CM8E2C 44460260 Ki = 154 nM T45262 CU8P5A 44460263 Ki = 244 nM T45262 CG12PW 44460272 Ki = 546 nM T45262 CBC95M 44460366 Ki > 10000 nM T45262 CU1K6W 44460367 Ki > 10000 nM T45262 CYW4E5 44460368 Ki = 514 nM T45262 C3VP6J 44460374 Ki > 10000 nM T45262 CIVL58 44460376 Ki > 10000 nM T45262 C6WLB3 44460545 Ki = 1002 nM T45262 C9Q8EA 44460546 Ki = 512 nM T45262 CH34CZ 44460553 Ki = 1035 nM T45262 C6UGE0 44460572 Ki = 370 nM T45262 C1QUL9 44460599 Ki = 338 nM T45262 CD3GB2 44460600 Ki = 330 nM T45262 COG5V3 44460602 Ki = 1066 nM T45262 CMT0E7 44462060 Ki = 190 nM T45262 C3YO4U 44462061 Ki = 1630 nM T45262 CC28UE 44462088 Ki = 7 nM T45262 CK1J3U 44462209 Ki = 620 nM T45262 C5Y0SX 44478733 IC50 = 63 nM T45262 C0G7FY 44543774 Ki = 14 nM T45262 C83MQV 44545161 Ki = 5 nM T45262 C48ULF 44545165 Ki = 0.373 nM T45262 C8E6CF 44545281 Ki = 91 nM T45262 CEKF72 44545284 Ki = 12 nM T45262 C35AVR 44545396 Ki = 7 nM T45262 CQ1FJ0 44587372 Ki = 1610 nM T45262 CJ1L7N 44587373 Ki = 76 nM T45262 CN1EL3 44587375 IC50 = 1 nM T45262 C5C2GS 44587376 Ki > 10000 nM T45262 CUA07D 44587377 Ki = 94 nM T45262 C2WY7R 44587378 Ki > 10000 nM T45262 CF9D0N 44587452 Ki = 561 nM T45262 C91ZPG 44587453 Ki = 277 nM T45262 CR95HX 44587454 Ki = 604 nM T45262 C5TH7B 44587455 Ki = 6 nM T45262 CS3Y2L 44587456 Ki = 8 nM T45262 C5FV4U 44587457 Ki = 9 nM T45262 C7FD5V 44587490 Ki = 33 nM T45262 CMB46A 44587491 Ki = 16 nM T45262 C12RQJ 44587492 Ki = 53 nM T45262 CP8O7G 44589092 IC50 = 27.54 nM T45262 CRM09K 44589115 IC50 = 58.88 nM T45262 C64EAP 44589202 IC50 = 87.1 nM T45262 CW2VX7 44589203 IC50 = 53.7 nM T45262 C4BS2N 44589204 IC50 = 100 nM T45262 CG71AO 44589205 IC50 = 128.82 nM T45262 CFA72S 44589206 IC50 = 162.18 nM T45262 C23LZI 44589221 IC50 = 3467.37 nM T45262 C19HTB 44589222 IC50 > 10000 nM T45262 C2JQ6I 44589223 IC50 = 257.04 nM T45262 C9M6RL 44589224 IC50 = 125.89 nM T45262 C4OUS0 44589236 IC50 = 173.78 nM T45262 C5LCO8 44589237 IC50 = 158.49 nM T45262 C9V5NG 44589238 IC50 = 56.23 nM T45262 C0UE2D 44589239 IC50 = 229.09 nM T45262 C6B8UC 44589256 IC50 = 2344.23 nM T45262 C3N6PV 44589257 IC50 = 851.14 nM T45262 CEI41U 44589258 IC50 = 7413.1 nM T45262 CU2RZ5 44589259 IC50 > 10000 nM T45262 CEL1M8 44589275 IC50 > 10000 nM T45262 CG0Q9F 44589276 IC50 > 10000 nM T45262 CNS86B 44589277 IC50 > 10000 nM T45262 CU80HV 44589278 IC50 = 3890.45 nM T45262 CFR07X 44589291 IC50 = 363.08 nM T45262 CLD0P4 44589302 IC50 = 34.67 nM T45262 CRD52K 44589303 IC50 = 8709.64 nM T45262 CK5UY1 44589304 IC50 = 2041.74 nM T45262 CX7Q6N 44589305 IC50 = 60.26 nM T45262 COWE29 44589306 IC50 = 213.8 nM T45262 CBN81E 44589317 IC50 = 158.49 nM T45262 C82JWG 44589318 IC50 = 89.13 nM T45262 C96OKQ 44589328 IC50 = 39.81 nM T45262 C4U0YH 44589329 IC50 = 257.04 nM T45262 CB39PO 44589330 IC50 = 363.08 nM T45262 CCWT68 44589331 IC50 = 223.87 nM T45262 C76HMO 44589348 IC50 = 93.33 nM T45262 CESC39 44589349 IC50 = 316.23 nM T45262 C04GPU 44589350 IC50 = 114.82 nM T45262 CU8XS0 44589351 IC50 = 144.54 nM T45262 CQI2A5 44593730 IC50 = 2 nM T45262 C64ALM 44610627 IC50 = 1.2 nM T45262 CQ49EP 45483574 IC50 = 1.9 nM T45262 C41TUO 45484976 Ki = 2500 nM T45262 C1OGA5 45484977 Ki = 132 nM T45262 CQR6S5 45484980 Ki = 43 nM T45262 CT19QL 45484981 Ki = 85 nM T45262 C9XMT6 45484988 Ki = 17 nM T45262 CGS15E 45484992 Ki = 183 nM T45262 C1QG3W 45485008 Ki = 577 nM T45262 C1IV6X 45485009 Ki = 135 nM T45262 CR4A9C 45485022 Ki = 117 nM T45262 COQ3H2 45485023 Ki = 193 nM T45262 CN0SR4 45485032 Ki = 129 nM T45262 C1YN6A 45485033 Ki = 1409 nM T45262 CGF3D5 45485034 Ki = 210 nM T45262 CQS6Y9 45485035 Ki = 76 nM T45262 C02ICQ 45485040 Ki = 13 nM T45262 C5U0JC 45485041 Ki = 996 nM T45262 CGM2T3 45485042 Ki = 574 nM T45262 CS71WM 45485045 Ki = 620 nM T45262 C0GUY3 45485050 Ki = 84 nM T45262 CZW07A 45485056 Ki = 124 nM T45262 C30FQC 45485057 Ki = 1130 nM T45262 CD86QS 45485064 Ki = 74 nM T45262 C1Z6MI 45485065 Ki = 101 nM T45262 CB21VP 45485073 Ki = 42 nM T45262 C4HPQ8 45485078 Ki = 632 nM T45262 C21BFH 45485079 Ki = 275 nM T45262 CD1VS8 45485080 Ki = 400 nM T45262 CCGQ13 45485086 Ki = 35 nM T45262 CWC67N 45485105 Ki = 32 nM T45262 CQB26E 46175148 Ki = 32 nM T45262 C4D1YH 46871760 Ki = 4.2 nM T45262 CC07VO 46872036 Ki = 3.9 nM T45262 CPS9D5 46872037 Ki = 4.4 nM T45262 CMS19X 46872038 Ki = 4.4 nM T45262 C8DE7N 46881383 Ki = 3300 nM T45262 CF6KS9 46881384 Ki > 5000 nM T45262 CFGW80 46881385 Ki > 5000 nM T45262 C4NS0C 46881386 Ki > 5000 nM T45262 CFI5L8 46881387 Ki > 5000 nM T45262 CL01JM 46881388 Ki > 5000 nM T45262 CFS5J4 46881389 Ki > 5000 nM T45262 C8CN5Y 46881390 Ki > 5000 nM T45262 C7HUS1 46881391 Ki > 5000 nM T45262 CL7EM0 46881392 Ki > 5000 nM T45262 C7BC1G 46881393 Ki > 5000 nM T45262 CPS93X 46881394 Ki > 5000 nM T45262 C7LQB5 46881395 Ki > 5000 nM T45262 C1UQ8L 46881396 Ki > 5000 nM T45262 CM3C9G 46881397 Ki = 19 nM T45262 C1C3KA 46881398 Ki = 1510 nM T45262 CU35LD 46881399 Ki > 5000 nM T45262 CS2RK7 46890768 Ki = 4800 nM T45262 CYX8R2 46890888 Ki = 4300 nM T45262 CPDC29 46890889 Ki = 1900 nM T45262 CRJC84 46890890 Ki = 7600 nM T45262 CG83NO 46890950 Ki = 1900 nM T45262 C6Y9JD 46890951 Ki > 7000 nM T45262 C6H1YB 46891008 Ki = 1200 nM T45262 CZ4P2U 46891009 Ki = 1600 nM T45262 C17FPY 46891010 Ki = 5800 nM T45262 C7NOR5 46891011 Ki = 3200 nM T45262 C1FA9U 46891057 Ki = 1700 nM T45262 C5KOY1 46891115 Ki = 470 nM T45262 CMX26E 46891116 Ki = 13 nM T45262 CE07PN 46891210 Ki = 16 nM T45262 CF9H7J 51352159 IC50 = 46 nM T45262 CG8X4M 52944875 Ki = 50.12 nM T45262 C49YVD 52947302 Ki = 25.12 nM T45262 C6RB2T 52947334 Ki = 50.12 nM T45262 C5T1IN 52947738 Ki = 79.43 nM T45262 C4LJK7 53309402 Ki = 68 nM T45262 CX8Q3F 53309547 Ki = 3657 nM T45262 C7B9PF 53309695 Ki = 27 nM T45262 C1OU5L 53310132 Ki = 7.2 nM T45262 CY6R4I 53310133 Ki = 4.2 nM T45262 C1VOH6 53310275 Ki = 7.6 nM T45262 C74TNR 53310276 Ki = 489 nM T45262 CK69EH 53310277 Ki = 26 nM T45262 C53FQE 53310410 Ki = 128 nM T45262 C0I5AH 54579975 IC50 = 3000 nM T45262 CA89OM 54579976 IC50 > 10000 nM T45262 CYM07O 54580961 IC50 = 970 nM T45262 C9U3PD 54580962 IC50 = 1600 nM T45262 CQ9IJ6 54580963 IC50 = 3100 nM T45262 C8Q6TC 54582017 IC50 = 7700 nM T45262 C1QS7N 54582962 IC50 = 3800 nM T45262 CA58BY 54585865 IC50 = 1100 nM T45262 C8BYX7 54585866 IC50 = 3000 nM T45262 COIC92 54586411 Ki = 4474 nM T45262 CLZ9G3 54586828 IC50 = 140 nM T45262 CH53NM 54586829 IC50 = 3300 nM T45262 CM94ZA 54586831 IC50 > 10000 nM T45262 CB30GL 54591779 Ki = 0.291 nM T45262 CRG91D 54591854 Ki = 19 nM T45262 C8IGE9 54754515 EC50 = 7.4 nM T45262 CZ40KM 54754516 EC50 = 8.6 nM T45262 CKF3H9 54754517 EC50 = 4.4 nM T45262 CK3E6D 56658150 Ki = 140 nM T45262 CG2V4C 56658860 Ki = 308 nM T45262 CEA3S5 56659877 EC50 = 234 nM T45262 C3SO6Z 56659947 IC50 = 42 nM T45262 CNWQ18 56659948 IC50 = 8 nM T45262 C2APK5 56659949 EC50 = 3.9 nM T45262 C2ZP0L 56661338 IC50 = 0.72 nM T45262 CI9LV3 56662342 Ki = 867 nM T45262 CN0QT9 56662343 Ki = 20 nM T45262 CM8UC3 56663335 EC50 = 95 nM T45262 CHV05I 56663336 EC50 = 97 nM T45262 CPJ4R7 56663337 IC50 = 76.7 nM T45262 CK52NJ 56663414 IC50 = 42 nM T45262 CI03BT 56663539 Ki = 103 nM T45262 CNZ68S 56665181 IC50 = 49 nM T45262 C2T0JZ 56666769 IC50 = 308 nM T45262 CWB2V7 56668206 IC50 = 30.6 nM T45262 CP2VR4 56668215 IC50 > 100 nM T45262 CXV6H7 56668632 IC50 = 3 nM T45262 C46WER 56668633 EC50 = 4 nM T45262 CO0V6N 56668634 EC50 = 8 nM T45262 CGZB32 56670201 EC50 = 75.7 nM T45262 CI1Y3T 56670270 EC50 = 58 nM T45262 C1X2EV 56670271 IC50 = 7.1 nM T45262 C0JZ4P 56672696 Ki = 607 nM T45262 CX7LB4 56672697 Ki = 11 nM T45262 CX0WL3 56672698 Ki = 9 nM T45262 C7P2ZL 56673724 EC50 = 53 nM T45262 CGI38W 56673725 IC50 = 13 nM T45262 CAJ06Z 56675099 IC50 > 100 nM T45262 CEW67U 56676057 Ki = 47 nM T45262 C7R8TM 56677028 EC50 = 113 nM T45262 C2N7TY 56677029 IC50 = 340 nM T45262 CG12ZA 56678852 IC50 = 6 nM T45262 CJ91NX 56680359 EC50 = 18.6 nM T45262 CSZ54K 56682683 Ki = 157 nM T45262 C84LPE 56682684 Ki = 261 nM T45262 CTF72G 56682685 Ki = 62 nM T45262 CY9Z6E 56683688 EC50 = 28.9 nM T45262 C43GVH 56683689 IC50 = 213 nM T45262 C9F6ZT 56683761 IC50 = 680 nM T45262 C1GN0X 56683762 EC50 = 889 nM T45262 CX03MT 56683763 EC50 = 46 nM T45262 C9O1UD 56683764 IC50 = 67 nM T45262 C5RSU3 56683765 IC50 = 20 nM T45262 CAF5Q2 56835112 Ki = 6 nM T45262 CERD56 56835113 Ki = 11 nM T45262 CLW4G9 57390211 EC50 = 47.2 nM T45262 CI6C0P 57390212 EC50 = 0.6 nM T45262 C60FTA 57390674 Ki = 52 nM T45262 CKI90H 57392001 EC50 = 1.2 nM T45262 C8F4VH 57393711 EC50 = 1.7 nM T45262 C6S3KI 57393712 IC50 = 122 nM T45262 C6F3IJ 57393713 EC50 = 1.1 nM T45262 CF57BU 57393714 EC50 = 5.5 nM T45262 CM45WI 57393715 IC50 = 131 nM T45262 CBP4S9 57395432 IC50 = 311 nM T45262 CPHF12 57395433 EC50 = 0.7 nM T45262 COD80V 57397276 EC50 = 1.2 nM T45262 C1N2QS 57397277 EC50 = 5.1 nM T45262 C5E7WA 57397278 EC50 = 3.7 nM T45262 COQ1E2 57397279 EC50 = 0.3 nM T45262 C0EA1I 57398970 EC50 = 3.5 nM T45262 C2D7UV 57398971 EC50 = 5 nM T45262 CDJ7G4 57398972 EC50 = 4.5 nM T45262 CT5PE0 57400679 EC50 = 4.2 nM T45262 CJ12GI 57400680 EC50 = 17.2 nM T45262 CVI37T 57400681 EC50 = 2.4 nM T45262 C7SLW0 57400682 EC50 = 1.1 nM T45262 C3P8AM 57400683 EC50 = 36.5 nM T45262 C1I6YH 57402455 EC50 = 7.4 nM T45262 CU2H9G 57402456 EC50 = 3.5 nM T45262 C87OBR 57785779 IC50 = 130 nM T45262 C9WX0G 57785808 IC50 = 210 nM T45262 CH8EX5 57785838 IC50 = 100 nM T45262 CPX1N0 57785862 IC50 = 11 nM T45262 C8IJH5 57786006 IC50 = 4.4 nM T45262 CKB89L 57786009 IC50 = 46 nM T45262 C94NJC 57786068 IC50 = 270 nM T45262 CL58WY 57786096 IC50 = 320 nM T45262 C7N3EZ 57786117 IC50 = 39 nM T45262 CL3Q1H 57786134 IC50 = 36 nM T45262 C4Z6PE 57786200 IC50 = 50 nM T45262 CZBW49 57786300 IC50 = 210 nM T45262 CC79KU 57786307 IC50 = 48 nM T45262 C0MA2T 57786312 IC50 = 20 nM T45262 CDH92T 57786313 IC50 = 66 nM T45262 COJ71I 57912441 IC50 = 98 nM T45262 CBF5R0 57912458 IC50 = 101 nM T45262 C96JRX 57912459 IC50 = 7.1 nM T45262 CUJ9Y3 58012303 IC50 = 7.9 nM T45262 CA18GJ 58012333 IC50 = 15 nM T45262 CS5GO9 58012370 IC50 = 7.4 nM T45262 CYJ6L5 58223382 IC50 = 61 nM T45262 CY7PX3 58223421 IC50 = 76 nM T45262 CL54PE 58223481 IC50 = 223 nM T45262 C3I5AG 58223502 IC50 = 48 nM T45262 CDW5J4 58730488 IC50 = 42 nM T45262 CGD31W 58801644 IC50 = 120 nM T45262 C7L6UG 58801647 IC50 = 120 nM T45262 C6BIE1 58801661 IC50 = 51 nM T45262 CWIB56 58801667 IC50 = 90 nM T45262 CC9O4Y 58896411 IC50 = 27 nM T45262 CC1Q5K 58896424 IC50 = 97 nM T45262 CRZH74 58896429 IC50 = 220 nM T45262 CUV71W 58896465 IC50 = 25 nM T45262 CX6W5D 58896474 IC50 = 14 nM T45262 CB48AC 58896475 IC50 = 990 nM T45262 C71CJB 58896512 IC50 = 90 nM T45262 C8WMB9 58896519 IC50 = 77 nM T45262 C3ZDM1 58896587 IC50 = 69 nM T45262 CZ8RA7 60141295 IC50 = 70 nM T45262 CYF35E 60155540 IC50 = 52 nM T45262 CIS4J2 60155541 Ki = 11 nM T45262 C7P1CR 60155708 IC50 = 22 nM T45262 CURH26 60155709 IC50 = 20 nM T45262 CA4U9W 60155710 IC50 = 40 nM T45262 CZQ18T 60155793 IC50 = 130 nM T45262 CZ46RJ 60155794 IC50 = 105 nM T45262 CA42RW 60155795 IC50 = 40 nM T45262 CF76GA 60155887 IC50 = 25 nM T45262 C1J9KM 60155888 IC50 = 47 nM T45262 CFIN43 60155889 IC50 = 98 nM T45262 C15ROB 60155989 IC50 = 27 nM T45262 CQD7X6 60155990 IC50 = 113 nM T45262 C8TR2N 60155991 IC50 = 34 nM T45262 CKEN80 60156090 IC50 = 194 nM T45262 C3VMJ6 68581422 IC50 = 84 nM T45262 CL4GB6 68581997 IC50 = 160 nM T45262 CY7QU4 70681899 IC50 = 646 nM T45262 CO67RY 70681900 IC50 = 157 nM T45262 C57HUT 70682070 IC50 = 197 nM T45262 CHK82U 70682293 IC50 = 70 nM T45262 C1X6ID 70682294 IC50 = 184 nM T45262 CH67UI 70684375 IC50 = 89 nM T45262 CV1Q9S 70684376 IC50 = 45 nM T45262 CI2WM3 70686154 IC50 = 323 nM T45262 CQ82EX 70686532 IC50 = 24 nM T45262 CWQ6U3 70686533 IC50 = 131 nM T45262 CT76XP 70688290 IC50 > 1000 nM T45262 C6F3LZ 70688432 IC50 = 88 nM T45262 CX0V3Z 70688433 IC50 = 75 nM T45262 CVCO30 70688637 IC50 = 246 nM T45262 CUF7L9 70688638 IC50 > 1000 nM T45262 C5CR8Z 70690301 IC50 = 762 nM T45262 CJMY25 70690480 IC50 = 742 nM T45262 C84CES 70690481 IC50 = 90 nM T45262 C16ZAP 70690703 IC50 = 212 nM T45262 CQ3BF7 70690704 IC50 = 23 nM T45262 CFU30R 70692469 IC50 = 79 nM T45262 C6NMB0 70692470 IC50 > 1000 nM T45262 CM6J1T 70692630 IC50 = 155 nM T45262 CZ98XI 70692631 IC50 = 100 nM T45262 C67FMV 70692632 IC50 = 672 nM T45262 C2K6GT 70692633 IC50 > 1000 nM T45262 CZJ38E 70692845 IC50 = 97 nM T45262 C1WVS4 70692846 IC50 = 88 nM T45262 CLW79I 70692847 IC50 = 286 nM T45262 CGHN83 70696576 IC50 = 138 nM T45262 CSJB53 70696577 IC50 > 1000 nM T45262 C9TK2Y 70696716 IC50 = 472 nM T45262 CCJU06 70696717 IC50 > 1000 nM T45262 CX1G6S 70696934 IC50 > 1000 nM T45262 CGPM10 70696935 IC50 = 375 nM T45262 CXR6D1 70696936 IC50 > 1000 nM T45262 CAO31E 70888282 IC50 = 1100 nM T45262 C6A8FP 70909662 IC50 = 110 nM T45262 C17ERF 70909665 IC50 > 10000 nM T45262 CBS51Y 70909803 IC50 = 170 nM T45262 CW71JY 70909805 IC50 = 9.5 nM T45262 C3E1IF 71449705 IC50 = 22 nM T45262 C0Z5RJ 71450106 IC50 = 75 nM T45262 C0K6SB 71451515 IC50 = 63 nM T45262 C0ZI4A 71451516 IC50 = 392 nM T45262 C2AK7S 71451919 IC50 = 69 nM T45262 CUM9S8 71451920 IC50 = 147 nM T45262 CZSM47 71453343 IC50 = 67 nM T45262 CD3C5H 71453344 IC50 = 57 nM T45262 CJF82U 71453426 Ki = 1.7 nM T45262 CM15IV 71453734 IC50 = 50 nM T45262 CQB82V 71453735 IC50 = 136 nM T45262 C09SAW 71453736 IC50 = 91 nM T45262 C5SQU2 71455050 IC50 = 28 nM T45262 CAO8U2 71455051 IC50 = 414 nM T45262 CBG2L1 71455052 IC50 = 75 nM T45262 CB0FZ9 71455053 IC50 = 65 nM T45262 CH6W7I 71455472 IC50 = 48 nM T45262 CBH6V7 71455473 IC50 = 46 nM T45262 CCR09G 71456848 IC50 = 43 nM T45262 CF0N9H 71456849 IC50 > 1000 nM T45262 CUV67I 71456850 IC50 = 91 nM T45262 CRTM90 71457262 IC50 = 65 nM T45262 C9ECA7 71457263 IC50 = 254 nM T45262 CW34DI 71458702 IC50 = 259 nM T45262 C3OJI8 71458703 IC50 = 36 nM T45262 CHCS73 71458704 IC50 = 202 nM T45262 CMIZ46 71458705 IC50 = 32 nM T45262 C5IL4B 71459110 IC50 = 126 nM T45262 CBOK19 71460919 IC50 = 83 nM T45262 C6TRY9 71462234 IC50 = 99 nM T45262 C6AXK5 71462615 IC50 = 43 nM T45262 CBG90L 73345508 IC50 > 100 nM T45262 CCVD49 73345509 IC50 > 500 nM T45262 CB65GT 73345736 Ki = 130 nM T45262 CS8D3J 73346924 IC50 = 24 nM T45262 C86PER 73348542 IC50 = 14 nM T45262 C32JUX 73348736 Ki > 1000 nM T45262 CXW60S 73348739 Ki = 48.9 nM T45262 C3I5TA 73348776 Ki = 1.07 nM T45262 C24WZC 73349901 IC50 = 18.4 nM T45262 C8UXB0 73350007 IC50 > 500 nM T45262 C1KJ7S 73350131 IC50 = 45 nM T45262 CZ9LY3 73350133 IC50 > 100 nM T45262 C75OIJ 73350317 Ki = 2 nM T45262 C61OBY 73351508 IC50 = 119 nM T45262 CDF4S9 73351515 IC50 = 10.2 nM T45262 CN3V9Y 73351613 IC50 > 100 nM T45262 C45OSY 73351614 IC50 > 100 nM T45262 CO1H4V 73351615 IC50 = 3.4 nM T45262 CZH5L2 73351616 IC50 = 5.9 nM T45262 CQ3FE7 73351824 Ki > 1000 nM T45262 CJ6MX9 73351827 Ki > 1000 nM T45262 CW12AB 73353094 IC50 = 7.7 nM T45262 C91IUQ 73353095 IC50 > 500 nM T45262 CV07PY 73353096 IC50 = 12 nM T45262 CG9U8K 73353098 IC50 = 1.9 nM T45262 C1OV4F 73354615 IC50 > 500 nM T45262 CLIJ68 73354788 EC50 = 3.5 nM T45262 CXJ6Q1 73354816 Ki = 44.8 nM T45262 CV18GL 73356172 IC50 > 100 nM T45262 CL78JX 73356174 IC50 = 0.24 nM T45262 C3KVB1 73356175 IC50 > 100 nM T45262 C59IAW 73356359 Ki = 50 nM T45262 C38JUH 73356364 Ki > 1000 nM T45262 C4P6FI 90231873 Ki = 1.3 nM T45262 C15TYE 90231885 Ki = 2.5 nM T45262 CRAZ42 90231888 Ki = 2.7 nM T45262 CP1BO8 90231897 Ki = 2.5 nM T45262 CYOD51 90654666 IC50 = 275.42 nM T45262 CQWX71 90654667 IC50 = 537.03 nM T45262 CC9Y0J 90654668 IC50 = 588.84 nM T45262 CO81SA 90654669 IC50 = 245.47 nM T45262 CBYR91 122193716 Ki = 3.4 nM T45262 C62JCT 122193717 Ki = 4.2 nM T45262 C0Z8CY 122193718 Ki = 4.4 nM T45262 CNS3J0 122193719 Ki = 5.4 nM T45262 CE63MF 122193720 Ki = 2.4 nM T45262 CJA01E 122193721 Ki = 180 nM T45262 C3JS4X 122193722 Ki = 16.4 nM T45262 CQXH97 122193723 Ki = 3.1 nM T45262 CHX1J0 122193724 Ki = 59 nM T45262 C2UH0X 122193725 Ki = 7.3 nM T45262 CB1K2A 122193726 Ki = 14.2 nM T45262 C4FGR1 122193727 Ki = 21.6 nM T45262 CPC10K 122193806 Ki = 13.9 nM T45262 CRVX74 127029856 Ki = 0.59 nM T45262 CUW08P 127029993 IC50 = 11 nM T45262 CG4LD7 127030304 IC50 = 22 nM T45262 CKF74S 127030314 IC50 = 24 nM T45262 CF9Y6N 127030336 IC50 = 140 nM T45262 CL1UD3 127030337 IC50 = 12 nM T45262 CJ4VA7 127030338 IC50 = 13 nM T45262 C4HO7M 127030634 IC50 = 2500 nM T45262 C9J0LZ 127030817 Ki = 0.61 nM T45262 CKJG94 127030922 IC50 = 2200 nM T45262 CK28ML 127030923 IC50 = 84 nM T45262 CHR08L 127030924 IC50 = 13 nM T45262 CF0BM3 127030925 IC50 = 7.6 nM T45262 CB7JF8 127030926 IC50 > 10000 nM T45262 CK68RO 127030927 IC50 = 13 nM T45262 CI1WG0 127031126 Ki = 0.69 nM T45262 CA4G3K 127031129 Ki = 0.52 nM T45262 CXV23A 127031132 Ki = 0.5 nM T45262 CCL04A 127031439 Ki = 0.34 nM T45262 CEYB78 127031441 Ki = 0.49 nM T45262 CAZ20H 127031514 IC50 = 14 nM T45262 CV23LT 127031736 Ki = 0.42 nM T45262 CD2CL7 127031738 Ki = 0.69 nM T45262 C9DN6B 127031741 Ki = 0.22 nM T45262 CS2MG6 127032010 Ki = 0.25 nM T45262 CS7VL0 127032314 Ki = 0.43 nM T45262 C4H0NM 127032315 Ki = 0.2 nM T45262 CO20BG 127033261 Ki = 0.81 nM T45262 CM8KB5 127033542 Ki = 0.18 nM T45262 CWAK93 127033544 Ki = 0.49 nM T45262 C8QKM7 127033836 Ki = 8.05 nM T45262 C6S0WC 127033837 Ki = 48.6 nM T45262 CE31AB 127033842 Ki = 0.24 nM T45262 C4QF2N 127033847 Ki = 0.68 nM T45262 CA0RX3 127033848 Ki = 0.74 nM T45262 CX7DB4 127034112 Ki = 48.98 nM T45262 C2BW3M 127053461 IC50 = 14 nM T45262 CXMV63 135553002 Ki = 930 nM T45262 C3ART6 135593026 Ki = 1181 nM T45262 C8PAH3 136000673 IC50 > 10000 nM T45262 CXD7O9 136029158 Ki = 560 nM T45262 C7QBJ8 136042277 EC50 = 688 nM T45262 C59GIP 136042278 EC50 = 4 nM T45262 C1G0FT 137635682 IC50 = 53 nM T45262 C4Q0AV 137635894 IC50 = 270 nM T45262 CW95DO 137640280 IC50 = 18 nM T45262 CGY0M3 137642541 IC50 = 150 nM T45262 C8KED6 137645497 Ki = 1.7 nM T45262 CI51GK 137646761 IC50 = 140 nM T45262 C2WQD1 137654892 IC50 = 110 nM T45262 C54FEV 137656239 IC50 = 48 nM T45262 C29IYF 137659453 Ki = 5 nM T45262 C6R7LQ 145948584 Ki = 5.94 nM T45262 CRU75L 145948590 Ki = 1.13 nM T45262 C9RAD4 145948591 Ki = 0.16 nM T45262 CJXE18 145948612 Ki = 0.7 nM T45262 CJS4D2 145948623 Ki = 0.53 nM T45262 CJC8Y4 145948644 Ki = 3 nM T45262 C1MGC8 145948645 Ki = 1.07 nM T45262 CB0ET7 145948680 Ki = 0.91 nM T45262 C0GE6W 145948692 Ki = 0.35 nM T45262 C6YVC5 145948693 Ki = 0.2 nM T45262 C3PN5A 145948700 Ki = 0.3 nM T45262 CK83OS 145948715 Ki = 0.29 nM T45262 CKU14Y 145948718 Ki = 0.45 nM T45262 CQ0EF3 145948720 Ki = 1.15 nM T45262 CO0KV7 145949031 Ki = 0.46 nM T45262 CIFS61 145955820 IC50 = 891.25 nM T45262 CBIP30 145958142 EC50 = 1.114 nM T45262 CSH53O 145959453 IC50 = 446.68 nM T45262 CLC76H 145967853 IC50 = 89 nM T45262 CL0YI3 145968300 IC50 = 18 nM T45262 CPTO89 145968888 IC50 = 350 nM T45262 CR13BY 145969226 IC50 = 55 nM T45262 C6HAJ3 145971087 IC50 = 200 nM T45262 C80YTG 155520133 IC50 = 580 nM T45262 CBUO17 155541854 IC50 = 75 nM T45262 CV1QA8 155543377 IC50 = 120 nM T45262 C4TR0C 155548925 IC50 = 69 nM T45262 CC91RM 155549579 IC50 = 50 nM T45262 CO02NX 155552287 IC50 = 25 nM T45262 C3TL1F 155553483 IC50 = 52 nM T45262 CQ2UO7 155561052 IC50 = 4400 nM T45262 C7L2KX 155561680 IC50 = 13 nM T45262 CKH7S3 155565844 IC50 = 53 nM T45262 CO60EV 155567202 IC50 = 1800 nM T45262 C9V4IY 155568703 IC50 = 120 nM T45262 C7MPZ2 10344587 Ki = 2 nM T45262 CH0V5Y 71462309 Ki = 1.7 nM T45262 D02IOC 5311055 Ki = 1.6 nM T45262 D04KWH 176157 Ki = 1.7 nM T45262 D06FIF 9862166 Ki = 12 nM T45262 D0C0AS 9800614 Ki = 5 nM T88185 D0N0ES 938 EC50 = 8.71 nM T88185 D0S1NZ 5310993 EC50 = 5300 nM T88185 D01DDN 56950369 EC50 = 2 nM T88185 D09TGC 49763030 EC50 = 12.9 nM T88185 D0A5MR 11159621 EC50 = 286 nM T88185 D0LI1C 44469321 IC50 > 10000 nM T88185 D0K1HO 51576 EC50 = 160 nM T88185 CWN03O 1047 EC50 = 6300 nM T88185 CJKY76 7420 EC50 = 215000 nM T88185 CBHG51 9822 EC50 = 24.55 nM T88185 CC2IU7 34037 EC50 = 368000 nM T88185 C28BJS 78346 EC50 = 2900 nM T88185 C4KL7M 88707 EC50 = 13600 nM T88185 CACL38 98845 EC50 = 500 nM T88185 CI53OT 120232 EC50 = 5300 nM T88185 CNXH01 231756 EC50 > 1000000 nM T88185 CR9G6U 247986 EC50 = 7600 nM T88185 CEN75C 643160 EC50 > 20000 nM T88185 CUB0S4 643402 Ki = 8100 nM T88185 C3WV2J 643403 Ki = 14000 nM T88185 CC7ZN1 735981 Ki = 5500 nM T88185 CW5A0Y 776416 Ki = 156 nM T88185 CDY49W 776464 EC50 = 100 nM T88185 CET1F4 853085 EC50 = 1300 nM T88185 C71SIN 882926 IC50 > 2500 nM T88185 CV6X3W 2734359 EC50 > 1000000 nM T88185 CK08WZ 2761046 EC50 = 23000 nM T88185 CY8JI4 2783146 EC50 > 1000000 nM T88185 C1FM0V 3159638 EC50 > 1000 nM T88185 CCI89O 4913402 EC50 = 79.43 nM T88185 CGJ90V 5358902 Ki = 410 nM T88185 C7W9XN 5369209 Ki = 180 nM T88185 CM4U8L 5475335 Ki = 760 nM T88185 CI3Q6P 5816396 Ki = 2500 nM T88185 C2RDU0 6057891 Ki = 4200 nM T88185 CQ58MB 6436431 Ki = 1000 nM T88185 C15ANE 6437229 Ki = 3500 nM T88185 CEFS70 7472024 EC50 > 1000000 nM T88185 C7NXL6 10103897 Ki = 700 nM T88185 CG9J8L 10197980 EC50 = 79.43 nM T88185 C1A5LT 11160694 EC50 = 1200 nM T88185 CO9SA3 11183317 IC50 = 4600 nM T88185 CNGR34 11183677 EC50 = 5000 nM T88185 CXG5D6 11183678 EC50 = 2400 nM T88185 CX3R0C 11184165 EC50 = 1100 nM T88185 CF5TN4 11206816 EC50 = 2000 nM T88185 C7T5ZM 11218626 EC50 = 2800 nM T88185 CE9H6X 11219885 EC50 = 4200 nM T88185 CCK36A 11228924 EC50 > 1000000 nM T88185 CSHA60 11264843 EC50 = 5400 nM T88185 C1PO6Q 11276453 EC50 = 480 nM T88185 CYLH85 11299550 IC50 = 2500 nM T88185 C6F1PI 11311474 EC50 = 2100 nM T88185 C2DAT1 11322738 EC50 = 1600 nM T88185 C4L1NT 11322761 EC50 = 12000 nM T88185 CG6T1I 11322762 EC50 = 6100 nM T88185 CO2TQ0 11323649 EC50 = 41000 nM T88185 CYA94T 11324121 EC50 = 740 nM T88185 CJ3S5D 11345283 EC50 = 5400 nM T88185 CA9B4T 11367769 EC50 = 46000 nM T88185 CPC18U 11368347 EC50 = 5700 nM T88185 CG2T6U 11379903 EC50 = 66 nM T88185 CM25BS 11380943 EC50 = 290 nM T88185 C3BGQ2 11390981 EC50 = 23000 nM T88185 C2W9MS 11413114 EC50 = 2500 nM T88185 C02QBE 11415838 EC50 = 7000 nM T88185 CHRK45 11424509 IC50 = 690 nM T88185 CJT29E 11446592 EC50 = 3700 nM T88185 CCXN52 11470032 EC50 = 33000 nM T88185 C1SJY0 11470798 EC50 = 7200 nM T88185 CS45ZG 11493732 IC50 = 21 nM T88185 C24AFH 11501164 IC50 = 87 nM T88185 CL4J9A 11501698 IC50 = 8 nM T88185 CSJ1L9 11508815 IC50 = 323 nM T88185 CDI7M3 11514051 EC50 = 14 nM T88185 C6ZG5T 11516324 EC50 = 34 nM T88185 C6CV5S 11516424 EC50 = 1100 nM T88185 CG8E3Q 11523095 EC50 = 1000 nM T88185 CQD54J 11523335 IC50 = 555 nM T88185 C2LK5Z 11550911 IC50 = 1700 nM T88185 CF8TD6 11557600 IC50 = 2200 nM T88185 C2RBZ7 11559598 IC50 = 283 nM T88185 CQJ54M 11560300 IC50 = 4 nM T88185 CF4B5X 11566404 IC50 = 120 nM T88185 CPJ4K9 11581300 IC50 = 86 nM T88185 CZ3GH6 11607970 EC50 = 27.5 nM T88185 C8QX1M 11610260 EC50 = 3400 nM T88185 C8J3BY 11610363 IC50 = 51 nM T88185 C0R1SW 11617480 EC50 = 86 nM T88185 CPS8R0 11617852 IC50 = 11 nM T88185 CN4CU6 11624691 IC50 = 16 nM T88185 C36MLA 11625092 EC50 = 120 nM T88185 CYL6Z3 11631886 IC50 = 940 nM T88185 CHDU46 11638560 IC50 = 34 nM T88185 CPV95E 11646179 IC50 = 18 nM T88185 CFR9P1 11646494 IC50 = 769 nM T88185 C56QYF 11647028 EC50 = 77 nM T88185 C26RUI 11658691 EC50 > 10000 nM T88185 CU53SD 11672831 EC50 = 1024 nM T88185 CTZW51 11693991 EC50 > 1000 nM T88185 CM4G2W 11710202 IC50 = 800 nM T88185 CD63TU 11736428 IC50 = 80 nM T88185 CB8YL0 11739420 EC50 = 430 nM T88185 CL7FM6 11817645 EC50 = 2600 nM T88185 CV7R8X 11845295 EC50 = 8300 nM T88185 C5U2WE 11852982 IC50 = 200 nM T88185 C8CRY2 11961288 EC50 > 10000 nM T88185 C85NVB 11992586 EC50 = 120.23 nM T88185 CXG82O 11992591 EC50 > 10000 nM T88185 C3ITV5 11992592 EC50 > 10000 nM T88185 C1QP5H 11992688 EC50 > 10000 nM T88185 CAV6P2 11992689 EC50 > 10000 nM T88185 C08TUH 11992692 EC50 > 10000 nM T88185 CS23KL 11992694 EC50 > 10000 nM T88185 CSK39Y 11992789 EC50 = 9332.54 nM T88185 CT5R7A 12002517 IC50 = 140 nM T88185 C3G8EU 12002518 IC50 = 70 nM T88185 CW7X8O 12002520 IC50 = 2700 nM T88185 CQ65OZ 12002521 IC50 = 7700 nM T88185 C9P2VQ 12002522 IC50 = 290 nM T88185 CYQ84H 12002523 IC50 = 1900 nM T88185 CFB57H 12002524 IC50 = 610 nM T88185 C68ERO 12002525 IC50 = 140 nM T88185 C7YPG9 12002616 IC50 = 760 nM T88185 CED30S 12002618 IC50 = 40 nM T88185 CXQ76S 12002619 IC50 = 2400 nM T88185 CA5KQ1 12002717 IC50 = 150 nM T88185 CE75DK 12002802 IC50 = 500 nM T88185 CU9OI3 12003490 IC50 = 20 nM T88185 C5M6KA 12003596 IC50 = 240 nM T88185 C4PF0A 12003597 IC50 = 90 nM T88185 CKL08Q 12003601 IC50 = 1900 nM T88185 C0D4WT 12003692 IC50 = 4000 nM T88185 CH8V4A 12003695 IC50 = 2100 nM T88185 C3J6XT 12003699 EC50 = 28000 nM T88185 C8C5XQ 12003785 IC50 = 270 nM T88185 CU2OC6 12003787 EC50 = 1100 nM T88185 C8Y3KE 12003788 IC50 = 220 nM T88185 CEPH65 12003790 IC50 = 460 nM T88185 C49LQV 12003791 IC50 = 600 nM T88185 C1T7CE 12003879 IC50 = 430 nM T88185 C2V1RW 12003880 IC50 = 410 nM T88185 CM2B0G 12430656 EC50 = 1500 nM T88185 C9CK5H 13071646 EC50 > 1000000 nM T88185 CU9J6V 13153555 Ki = 72 nM T88185 CVZR52 14112183 Ki = 5700 nM T88185 C5ZQ9X 15604637 EC50 = 4 nM T88185 C4HW0N 15604638 EC50 = 10 nM T88185 CWN02L 15604641 EC50 = 5 nM T88185 CV3WB0 15604642 EC50 = 4 nM T88185 CN5L4Q 15604644 EC50 = 26 nM T88185 CM2NE9 15605287 EC50 = 31 nM T88185 CIOL71 15605292 EC50 = 930 nM T88185 CR6X0G 15605357 EC50 = 1300 nM T88185 CG17ZD 15605359 EC50 = 425 nM T88185 C1GD7L 15605364 EC50 = 285 nM T88185 C0YR6A 15605498 EC50 = 133 nM T88185 CG47KX 15605500 EC50 > 10000 nM T88185 CZJ2A1 15605503 EC50 = 738 nM T88185 CE7IR0 15605571 EC50 = 17 nM T88185 C26RYI 15605645 EC50 = 19 nM T88185 CGW36A 15605646 EC50 = 28 nM T88185 C3TZO1 15605648 EC50 = 10 nM T88185 CE5FG1 15605654 EC50 = 13 nM T88185 CE3W1R 15735511 EC50 > 1000000 nM T88185 C21HBP 15981408 EC50 = 9100 nM T88185 C93AMQ 15986754 EC50 = 8300 nM T88185 CNXM59 15986755 EC50 = 76 nM T88185 C0DWJ8 15986929 IC50 = 26 nM T88185 CR9FH7 15986930 EC50 = 620 nM T88185 CEMJ79 15986931 IC50 = 5 nM T88185 CX37OI 15986936 EC50 = 200 nM T88185 C67UCM 16048768 IC50 = 650 nM T88185 C7DS2N 16048770 IC50 = 550 nM T88185 C4GI5X 16048839 IC50 = 1200 nM T88185 CILM98 16048840 EC50 = 4600 nM T88185 C97OXR 16048843 EC50 = 17000 nM T88185 CZ5SO7 16048845 EC50 = 7900 nM T88185 CRP0C3 16048917 EC50 = 11000 nM T88185 CB1K6W 16048919 IC50 = 290 nM T88185 CJ4PI6 16048921 IC50 = 5700 nM T88185 C7E6RZ 16048923 IC50 = 2200 nM T88185 CM5L3O 16048992 IC50 = 2100 nM T88185 C6PTJ0 16048993 EC50 = 7800 nM T88185 CH41OM 16048995 EC50 = 13000 nM T88185 C1SX6J 16048997 IC50 = 20000 nM T88185 CQ4FA9 16048998 EC50 = 5900 nM T88185 CH9MY5 16124880 EC50 > 50000 nM T88185 C4R2DP 16125019 EC50 > 50000 nM T88185 C3F4KP 16125020 EC50 = 19000 nM T88185 C24KGF 16125021 EC50 > 100000 nM T88185 C6O5CE 17688981 EC50 > 1000 nM T88185 CQ8CF5 17751630 IC50 = 28 nM T88185 C0VYB1 17925840 EC50 = 6100 nM T88185 CIX0N5 19359201 EC50 > 1000000 nM T88185 CJYU53 21660892 EC50 > 1000 nM T88185 C73XOY 21798667 EC50 > 1000000 nM T88185 CH7XV6 22052341 EC50 > 1000000 nM T88185 C3L5WA 24180571 EC50 = 41.69 nM T88185 CF6XS1 24741208 EC50 > 20000 nM T88185 C5T7EA 24741306 IC50 = 350 nM T88185 CIAV47 24741307 EC50 = 93 nM T88185 C1KQI0 24741310 IC50 = 58 nM T88185 CM4HE6 24741312 EC50 = 240 nM T88185 CVKT72 24811199 EC50 = 410 nM T88185 CI15FQ 24811547 IC50 = 34 nM T88185 CX37FW 24811550 EC50 = 64 nM T88185 CCQ0L8 24953853 EC50 = 67 nM T88185 C5IF6G 24953854 EC50 = 22 nM T88185 C4ZXS6 24953855 EC50 = 66 nM T88185 CPQJ96 24953857 EC50 = 172 nM T88185 CM91XK 24954201 EC50 = 90 nM T88185 C27ETC 24954204 EC50 = 128 nM T88185 CJ2I4U 24954566 EC50 = 1402 nM T88185 CA89OI 24954572 EC50 = 179 nM T88185 C30CJH 24954935 EC50 = 53 nM T88185 CB5TL0 24954940 EC50 = 137 nM T88185 CE84GT 24954941 EC50 = 108 nM T88185 C8V4OP 24955288 EC50 = 245 nM T88185 CAO68S 24955289 EC50 > 10000 nM T88185 C98CVD 24955294 EC50 = 451 nM T88185 CDQ92B 24955642 EC50 = 308 nM T88185 CDQK67 24955646 EC50 = 49 nM T88185 C7D6YH 28400046 EC50 = 35000 nM T88185 CR2F3V 28400056 EC50 = 20000 nM T88185 C73LBP 42625213 EC50 = 690 nM T88185 C2H6QR 42625218 IC50 = 6 nM T88185 CJPW47 42625379 IC50 = 3 nM T88185 CLPU71 42625380 IC50 = 360 nM T88185 CW7A0V 42625382 IC50 = 340 nM T88185 CT0H2G 42625474 IC50 = 3 nM T88185 CGI02C 42625475 IC50 = 1 nM T88185 CS34QO 42625476 IC50 = 1 nM T88185 CO2MW3 44351665 EC50 = 2700 nM T88185 CNO80I 44433524 EC50 = 57.54 nM T88185 CFH9B5 44433525 EC50 = 269.15 nM T88185 CH23EV 44433526 EC50 > 1000 nM T88185 C5B1MV 44433527 EC50 > 1000 nM T88185 CIV5T0 44433528 EC50 > 1000 nM T88185 C4GC8E 44433529 EC50 > 1000 nM T88185 CJQP40 44433530 EC50 > 1000 nM T88185 C5QKD9 44433531 EC50 > 1000 nM T88185 CWJ8H0 44433532 EC50 = 758.58 nM T88185 C02HSO 44433533 EC50 > 1000 nM T88185 CMK49L 44433534 EC50 > 1000 nM T88185 CC1UV3 44441302 EC50 > 1000 nM T88185 C78QVW 44441304 EC50 = 8700 nM T88185 C6L1SG 44441305 EC50 = 4900 nM T88185 C46XHD 44441310 EC50 = 12200 nM T88185 CV0AS8 44441311 EC50 = 2500 nM T88185 CW1GA3 44441312 EC50 = 5600 nM T88185 CTB83Y 44441316 EC50 = 6600 nM T88185 CF1S3H 44441318 EC50 = 12000 nM T88185 C2Q9IP 44441320 EC50 = 2500 nM T88185 C4R9WC 44441321 EC50 = 8700 nM T88185 C3HF4G 44441322 EC50 = 2100 nM T88185 C2FMP9 44441323 EC50 = 5600 nM T88185 C3VM4X 44441326 EC50 = 2200 nM T88185 C9W6MH 44445341 EC50 = 6300 nM T88185 C3XJ1K 44579645 EC50 = 930 nM T88185 CHLX51 44579646 EC50 = 1800 nM T88185 CYJ64R 44579647 EC50 = 460 nM T88185 CCIK12 44579648 EC50 = 2300 nM T88185 C8SP4O 44579693 EC50 = 1300 nM T88185 C5H3PA 44579742 EC50 = 940 nM T88185 CT5O3Q 44579761 EC50 = 2100 nM T88185 CG6O0B 44579762 EC50 = 700 nM T88185 CT8V5E 44579763 EC50 = 3000 nM T88185 CBD15I 44579779 EC50 = 1900 nM T88185 C47KQC 44579780 EC50 = 1400 nM T88185 C2J0XB 44580007 EC50 = 3200 nM T88185 C41KFD 44580008 EC50 = 6000 nM T88185 C5OYG8 44580036 EC50 = 2300 nM T88185 C89LVM 44580038 EC50 = 1300 nM T88185 CI07TR 44591586 IC50 = 4800 nM T88185 CP9QU1 44591601 IC50 = 870 nM T88185 CB5LX3 44591602 IC50 = 5200 nM T88185 CH8NZ7 44591603 IC50 = 16000 nM T88185 C7LDW4 44591604 IC50 = 5000 nM T88185 C0M9VC 45267309 EC50 > 10000 nM T88185 CSQ82F 45269046 EC50 > 10000 nM T88185 CJC95S 45269912 EC50 > 10000 nM T88185 C71YHO 45269913 EC50 > 10000 nM T88185 CVCP51 45270725 EC50 > 10000 nM T88185 C0R9FC 45271541 EC50 > 10000 nM T88185 C1HFL2 45272461 EC50 > 10000 nM T88185 CHKO74 46889319 EC50 = 45 nM T88185 COL87W 46889320 EC50 = 2350 nM T88185 COLU28 46889336 EC50 = 244 nM T88185 CK20GZ 46889337 EC50 = 504 nM T88185 CKT4V2 46889338 EC50 = 1110 nM T88185 CP30MX 46889339 EC50 = 156 nM T88185 CM7U5I 46889340 EC50 = 507 nM T88185 CKSO17 46889341 EC50 = 541 nM T88185 CXO84F 46889342 EC50 = 276 nM T88185 CFS5E3 46889360 EC50 = 12900 nM T88185 CUQG02 46889361 EC50 = 1420 nM T88185 C8RHE1 46889362 EC50 = 23100 nM T88185 CGW2H1 46889363 EC50 = 2450 nM T88185 C19EGN 46889364 EC50 = 3750 nM T88185 CW14ZG 46889397 EC50 = 1830 nM T88185 CP05MB 46889398 EC50 = 2860 nM T88185 C87GFP 46889399 EC50 = 2000 nM T88185 C3C7OD 46890163 EC50 = 9500 nM T88185 CWSN39 46890164 IC50 = 260 nM T88185 CRXN82 46890165 EC50 = 340 nM T88185 C4LB5U 46890197 EC50 = 940 nM T88185 C71SKI 46890198 EC50 = 750 nM T88185 CW2XE5 46890199 EC50 = 3000 nM T88185 CS87DX 46890237 EC50 = 280 nM T88185 C1Z4CG 46890238 EC50 = 770 nM T88185 C24GDK 46890239 IC50 = 22 nM T88185 CQ53DS 46890240 IC50 = 5 nM T88185 CK2YT3 46890268 EC50 = 430 nM T88185 C97PDE 46890269 IC50 = 8 nM T88185 CB9NU1 46890270 IC50 = 6 nM T88185 CQ8F4G 46890271 IC50 = 420 nM T88185 CZ7W0Y 46890272 EC50 = 370 nM T88185 CA2YM6 46890273 IC50 = 1310 nM T88185 CURT34 46890274 EC50 = 170 nM T88185 CE69AX 46890275 EC50 = 130 nM T88185 CG45JB 46890276 EC50 = 230 nM T88185 C7AV1Q 46890296 EC50 = 5300 nM T88185 CD0G7H 46890297 IC50 = 11 nM T88185 CC4NU5 46890298 IC50 = 7.4 nM T88185 CEGQ73 46890299 EC50 = 130 nM T88185 C0LKY1 46890300 IC50 = 6 nM T88185 CVAU45 46890301 IC50 = 5 nM T88185 CHRI47 46890302 EC50 = 95 nM T88185 C9P1HZ 46890327 EC50 = 11 nM T88185 C2OR8D 46890328 EC50 = 94 nM T88185 C87MIF 46890399 IC50 = 14 nM T88185 C7UQM5 46890400 EC50 = 2650 nM T88185 C1L0XQ 46890401 IC50 = 36 nM T88185 CG5LK1 46890500 IC50 = 35 nM T88185 CFXE41 46890501 IC50 = 32 nM T88185 CJ42TG 46890537 EC50 = 230 nM T88185 CFM43L 46890538 IC50 = 85 nM T88185 C0Z8MP 46890539 EC50 = 22 nM T88185 CFS19N 46890577 EC50 = 45 nM T88185 CHDZ10 46890578 EC50 = 46 nM T88185 CTLE08 46890579 EC50 = 7400 nM T88185 CNLO62 46890580 IC50 = 6 nM T88185 CBL3O2 49862072 IC50 = 380 nM T88185 CBF2W6 49862073 IC50 = 1700 nM T88185 C0UW3M 49862074 IC50 = 1300 nM T88185 CGW84J 51346919 EC50 = 59 nM T88185 C2EM4H 52941721 IC50 = 150 nM T88185 CH0U9I 52947887 EC50 = 2300 nM T88185 CJ9X1E 52947888 EC50 = 1100 nM T88185 CZE7B8 53224766 EC50 > 1000000 nM T88185 C6Q2MA 53317449 EC50 = 1110 nM T88185 C8PG4J 53317467 EC50 = 3119 nM T88185 CGX71J 53317490 EC50 > 10000 nM T88185 CXLW41 53317491 EC50 = 821 nM T88185 C85OZQ 53317492 EC50 = 379 nM T88185 CUL45B 53317493 EC50 > 10000 nM T88185 CDF7Z1 53318725 EC50 > 10000 nM T88185 CU0Q8O 53318740 EC50 = 6065 nM T88185 CTB29G 53318741 EC50 = 4436 nM T88185 C9Z3IF 53318746 EC50 = 327 nM T88185 CI6BZ3 53318768 EC50 = 353 nM T88185 C25BNY 53320057 EC50 > 10000 nM T88185 C8RPJ2 53320337 EC50 > 10000 nM T88185 C7G0QU 53321350 EC50 > 10000 nM T88185 C5OXD9 53321351 EC50 > 10000 nM T88185 CU7Q4W 53321367 EC50 = 6581 nM T88185 C3HBQ5 53321368 EC50 = 4152 nM T88185 C4FPK7 53321396 EC50 = 479 nM T88185 CV0LY9 53322689 EC50 = 470 nM T88185 C09UWM 53322717 EC50 = 130 nM T88185 C1HDF4 53324022 EC50 = 2705 nM T88185 CA54WP 53324023 EC50 > 10000 nM T88185 C7PGM2 53324024 EC50 = 275 nM T88185 CO9S6G 53324025 EC50 > 10000 nM T88185 CIF95V 53324033 EC50 = 3108 nM T88185 C8JGC7 53324034 EC50 = 787 nM T88185 CL2HW5 53324057 EC50 = 591 nM T88185 CO9JH1 53325308 EC50 > 10000 nM T88185 CQMR64 53325309 EC50 = 3393 nM T88185 CP0AI3 53325342 EC50 = 1076 nM T88185 CPL5V3 53325627 EC50 > 10000 nM T88185 CV58FJ 53326574 EC50 > 10000 nM T88185 CY8D3L 53326575 EC50 > 10000 nM T88185 CE6ID7 53326590 EC50 > 10000 nM T88185 CC3NG2 53326591 EC50 = 281 nM T88185 COW39R 53326616 EC50 = 335 nM T88185 CYM94U 53326893 EC50 = 1261 nM T88185 C4EUP6 54580649 Ki = 10000 nM T88185 CF9C7B 54580748 IC50 = 13 nM T88185 CF54NB 54582648 Ki = 9800 nM T88185 CPV94K 54582649 Ki = 2400 nM T88185 CZ50JU 54583606 Ki = 8900 nM T88185 CV7F4T 54584718 IC50 = 21 nM T88185 CP2B9Y 54585613 EC50 = 1000 nM T88185 CS05JP 54587625 IC50 = 150 nM T88185 CT1X5U 56659539 EC50 = 380 nM T88185 CQT70V 56950649 EC50 = 63 nM T88185 CY0K8Q 57390147 EC50 = 319 nM T88185 C4DFE0 57390148 EC50 = 238 nM T88185 CK8PH6 57390149 EC50 = 312 nM T88185 CAY03I 57391931 EC50 = 588 nM T88185 CL61JH 57391932 EC50 = 911 nM T88185 CJ4WY8 57392461 EC50 = 1388 nM T88185 CJK9M1 57393654 EC50 = 125 nM T88185 C6H7YF 57393655 EC50 = 138 nM T88185 C8C2BR 57393656 EC50 = 260 nM T88185 CF2UN7 57395376 EC50 = 113 nM T88185 C69UOR 57395377 EC50 = 96 nM T88185 C2OW6X 57397199 EC50 = 190 nM T88185 CYJ3K7 57397200 EC50 = 10000 nM T88185 CS03JM 57397201 EC50 = 1061 nM T88185 C6FXZ4 57397202 EC50 = 723 nM T88185 C30IQD 57397203 EC50 = 424 nM T88185 CY9JZ7 57397204 EC50 > 1000 nM T88185 CX9YK3 57398904 EC50 = 2060 nM T88185 C02VCJ 57398905 EC50 = 860 nM T88185 CKL03G 57398906 EC50 = 34 nM T88185 CJ0Z2N 57400594 EC50 = 290 nM T88185 C6UZW2 57400595 EC50 = 270 nM T88185 C30RQB 57400596 EC50 = 93 nM T88185 CT9PW5 57400597 EC50 = 10000 nM T88185 CPW74O 57400598 EC50 = 177 nM T88185 CDA29Y 57400599 EC50 = 26 nM T88185 CUHD29 57402396 EC50 = 10000 nM T88185 CC8H3K 57402397 EC50 = 417 nM T88185 CZ3I9R 57402398 EC50 = 291 nM T88185 C6MFY9 57402399 EC50 > 1000 nM T88185 C4NG8S 57412208 EC50 > 10000 nM T88185 CG2DI8 57412209 EC50 > 10000 nM T88185 C15WGL 57412210 EC50 = 1170 nM T88185 C5LCE9 57412211 EC50 = 21280 nM T88185 C03UIR 57412214 EC50 = 311 nM T88185 CHMG16 57412216 EC50 = 22.5 nM T88185 CT8ON4 57412217 EC50 = 1630 nM T88185 CCM57T 57412218 EC50 = 5450 nM T88185 C24LCT 57412296 EC50 > 10000 nM T88185 CR37YI 57412297 EC50 = 5330 nM T88185 C1YX8S 57412298 EC50 > 10000 nM T88185 C6L1NJ 57412299 EC50 > 10000 nM T88185 C03IQT 57412300 EC50 = 227 nM T88185 CHC8V0 57412301 EC50 = 7.4 nM T88185 CPNZ32 57412302 EC50 = 2470 nM T88185 C6XVF9 57412303 EC50 = 857 nM T88185 CK4PM0 57412304 EC50 > 10000 nM T88185 CU7GH8 57412400 EC50 = 276 nM T88185 C5RZ8G 57413367 EC50 = 16.4 nM T88185 C97WCF 57413446 EC50 = 1770 nM T88185 CX53ZS 57413447 EC50 = 225 nM T88185 CJO41C 57413448 EC50 = 1120 nM T88185 CC0VJ9 57413450 EC50 = 81 nM T88185 C0TY6F 57413451 EC50 > 10000 nM T88185 CRD2S4 57413453 EC50 = 1290 nM T88185 CBK2A5 57413541 EC50 = 28 nM T88185 C3I7ZJ 57413542 EC50 = 1980 nM T88185 C9GZ3K 57413544 EC50 = 141 nM T88185 CG89NH 57413545 EC50 = 83 nM T88185 CSD3Y0 57413546 EC50 = 192 nM T88185 CJS6P7 57413547 EC50 > 10000 nM T88185 C0YXZ2 59304594 EC50 = 47 nM T88185 CEDC82 59304608 EC50 = 1 nM T88185 CM2JN8 59304624 EC50 = 99 nM T88185 CV02UG 59304655 EC50 = 110 nM T88185 CL21IS 59304795 EC50 = 290 nM T88185 C03CTR 59304808 EC50 = 1600 nM T88185 C79NIK 59304857 EC50 > 10000 nM T88185 C14MRY 59304859 EC50 = 470 nM T88185 CFU50D 59304931 EC50 = 220 nM T88185 CS4RK1 59304946 EC50 = 11 nM T88185 C7O0MY 59304949 EC50 = 230 nM T88185 C23VNR 59304954 EC50 = 39 nM T88185 C74AYK 59343597 EC50 = 7 nM T88185 CD2K5L 59343651 EC50 = 16 nM T88185 CF70SZ 59343664 EC50 = 3 nM T88185 C89RDH 66560365 EC50 > 1000000 nM T88185 CX5K1I 66560366 EC50 > 1000000 nM T88185 C4VB8Y 66560367 EC50 > 1000000 nM T88185 CMQB78 70681781 EC50 = 170 nM T88185 CNY87V 70683894 EC50 = 6100 nM T88185 CBT14E 70683908 EC50 = 16 nM T88185 CLTD28 70686030 EC50 > 10000 nM T88185 C4G5OK 70686047 EC50 = 310 nM T88185 C07HZI 70686422 EC50 > 10000 nM T88185 CNP70F 70688150 EC50 > 10000 nM T88185 C42IAY 70696472 EC50 > 10000 nM T88185 CU3QF4 90645401 EC50 = 1400 nM T88185 CFS18J 90645402 EC50 = 900 nM T88185 C7RDB4 90645403 EC50 = 4500 nM T88185 C59MSV 90645404 EC50 = 4100 nM T88185 C4E2HW 90645405 IC50 = 327 nM T88185 CT1G5Y 90645406 EC50 = 4100 nM T88185 CHA60M 90645407 EC50 = 27400 nM T88185 CUS5N3 90645408 EC50 = 6800 nM T88185 C2B4XI 90645409 EC50 = 6300 nM T88185 CP3AR8 90645410 EC50 = 5800 nM T88185 C1T7SY 90645411 EC50 = 51600 nM T88185 C2E7IW 90645412 EC50 = 26300 nM T88185 CLN13S 90645413 EC50 = 12500 nM T88185 CA3X8J 90645414 EC50 = 36400 nM T88185 CKET69 122181102 IC50 = 1401 nM T88185 C6H2DV 122181103 IC50 = 83 nM T88185 CCGE32 122181104 IC50 = 326 nM T88185 CV1SP5 122181105 IC50 = 201 nM T88185 C3NRX7 122181106 IC50 = 365 nM T88185 CNI0B2 122181107 IC50 = 91 nM T88185 C2I1GZ 122181139 IC50 = 129 nM T88185 C3Y9TH 122181140 IC50 = 23 nM T88185 CC48UH 122181141 IC50 = 58 nM T88185 C6FY3T 122181142 IC50 = 21 nM T88185 C7PHA2 122181143 IC50 = 105 nM T88185 C06JYZ 135399731 IC50 = 35 nM T88185 CP6CZ4 135401973 EC50 = 470 nM T88185 C4XC6P 135401974 IC50 = 870 nM T88185 C4H8GO 135401975 EC50 = 5800 nM T88185 C7D6WK 135416383 IC50 = 13 nM T88185 CX1UD2 135416384 IC50 = 4 nM T88185 COQA52 135416388 Ki = 3 nM T88185 CP4B5A 135416391 Ki = 29 nM T88185 CT9Q8F 135416392 Ki = 4 nM T88185 C7NY5Q 135416393 Ki = 22 nM T88185 CRY8Q1 135453098 IC50 = 1 nM T88185 CB1M4T 135466520 EC50 = 50 nM T88185 CWGT82 135502978 EC50 = 74 nM T88185 C7W8HO 135627640 IC50 = 100 nM T88185 C3KD4S 135800175 IC50 = 330 nM T88185 C01PRA 135800176 IC50 = 26 nM T88185 CC69TI 135800177 IC50 = 10 nM T88185 C62NHL 135800194 Ki = 4 nM T88185 C7C9RS 135812996 IC50 = 450 nM T88185 C3DM1J 135887285 Ki = 11 nM T88185 CNC07T 135887288 Ki = 360 nM T88185 CA2K4M 135887289 Ki = 130 nM T88185 C8JSW3 135887290 Ki = 1.4 nM T88185 C9TI0R 135899108 IC50 = 1200 nM T88185 CKWQ06 135899109 IC50 = 4300 nM T88185 CV8GX7 135899110 IC50 = 4400 nM T88185 CI76OA 135899129 IC50 = 1100 nM T88185 C1V6NZ 135899130 IC50 = 4700 nM T88185 C5AUT3 135899131 IC50 = 250 nM T88185 CB7SM5 135899149 IC50 = 370 nM T88185 CA86ER 135899150 IC50 = 860 nM T88185 C2W5CZ 135899152 IC50 = 1700 nM T88185 C34WRL 135899153 IC50 = 440 nM T88185 C5C4KO 135899154 IC50 = 600 nM T88185 CQW09D 135899170 IC50 = 230 nM T88185 C2K3QR 135899171 IC50 = 15 nM T88185 CLM28F 135899178 IC50 = 50 nM T88185 CQ0D2M 135899198 IC50 = 230 nM T88185 C9GI4S 135899199 IC50 = 1500 nM T88185 C2J0DU 135899244 IC50 = 5900 nM T88185 C4RGN6 135899259 IC50 > 50000 nM T88185 C6EU5B 135899280 IC50 = 920 nM T88185 CT2K0S 135899300 IC50 = 840 nM T88185 CNG32A 135899320 IC50 = 130 nM T88185 CMW7U4 135899321 IC50 = 670 nM T88185 CCP37R 135899322 IC50 = 220 nM T88185 CJOU12 135899324 IC50 = 6300 nM T88185 CC52JR 135899325 EC50 = 2500 nM T88185 C5SAI0 135922719 IC50 = 2100 nM T88185 CJ41MZ 135922722 IC50 = 130 nM T88185 CUX64Z 135922723 IC50 = 380 nM T88185 CB8H5Q 135966934 EC50 = 27 nM T88185 C6WT2Z 136000579 IC50 = 42 nM T88185 CO7K3C 136000580 EC50 = 85 nM T88185 CA5O7N 136000619 EC50 < 52 nM T88185 CBC64N 136000669 EC50 = 1500 nM T88185 C18BPF 136000718 IC50 = 108 nM T88185 CSJC85 136086823 EC50 = 17 nM T88185 CKS53C 136086824 EC50 = 98 nM T88185 C3D8VI 136086828 EC50 = 6 nM T88185 CAT74E 136086829 EC50 = 42 nM T88185 CK1YO0 136088957 EC50 = 3420 nM T88185 CNM8O5 136088958 EC50 = 36 nM T88185 C9ZK4U 136088959 IC50 = 100 nM T88185 C49KYR 136088960 EC50 = 39 nM T88185 C31DJN 136088961 EC50 = 721 nM T88185 C3WO1Y 136088962 IC50 = 41 nM T88185 C5MGD1 136127010 IC50 = 1300 nM T88185 CWZ16U 136127011 IC50 > 50000 nM T88185 C8L6AT 136127012 IC50 = 48000 nM T88185 CVH9E8 136127013 IC50 > 50000 nM T88185 CD78CP 136127014 IC50 > 50000 nM T88185 CCK0A2 136127016 IC50 = 33 nM T88185 C3OD8Q 136127017 IC50 = 410 nM T88185 C8TE1P 137632012 IC50 = 37 nM T88185 CLI6E3 137633734 IC50 = 25 nM T88185 C5G8RH 137635325 IC50 = 13 nM T88185 C0UZ8L 137635425 IC50 = 28 nM T88185 CN0T1Y 137637662 IC50 = 58 nM T88185 C80DYL 137639493 EC50 = 36 nM T88185 CC7P6F 137640776 IC50 = 16 nM T88185 CO5YN6 137641317 EC50 = 130 nM T88185 CQ28VJ 137645601 IC50 = 2828 nM T88185 C7UF1G 137647495 IC50 = 32 nM T88185 C7ICD4 137648318 IC50 = 3620 nM T88185 CY2ID7 137648386 EC50 = 9 nM T88185 CXQH91 137650474 IC50 = 40 nM T88185 C4MS6X 137652577 EC50 = 110 nM T88185 CFW89L 137653026 EC50 = 270 nM T88185 CH6PL9 137653428 EC50 = 630 nM T88185 C8DP3Y 137654580 EC50 = 390 nM T88185 C3DNK2 137655320 IC50 = 138 nM T88185 COY5K3 137659759 IC50 = 665 nM T88185 CM0WT4 137661033 IC50 = 229 nM T88185 CW8JC3 137661636 IC50 = 56 nM T88185 CKVQ61 137662135 EC50 = 190 nM T88185 C35EKW 145949989 EC50 = 30.48 nM T88185 COBH03 145954324 EC50 = 1005 nM T88185 C6F5HC 145957123 EC50 = 454 nM T88185 CDF90G 145957566 EC50 = 10.59 nM T88185 CL1H7R 145960556 EC50 = 275.42 nM T88185 D00TPG 11041813 EC50 = 8900 nM T88185 D01AUX 11617151 IC50 = 94 nM T88185 D02GRY 11148966 EC50 = 24000 nM T88185 D02YVZ 135899263 IC50 = 19000 nM T88185 D05VGC 53238781 EC50 = 214 nM T88185 D06UZK 648852 Ki = 3500 nM T88185 D06WXN 12003694 IC50 = 390 nM T88185 D07BFA 4268702 EC50 = 1200 nM T88185 D07NDW 25101223 EC50 = 120 nM T88185 D07ONY 11776293 IC50 = 4200 nM T88185 D07TVE 11672811 EC50 = 210 nM T88185 D07XKG 135899247 IC50 = 4400 nM T88185 D08ZYC 11595431 EC50 < 6309.57 nM T88185 D09ZPN 135416394 Ki = 4 nM T88185 D0AU0M 637542 Ki = 14000 nM T88185 D0ET2F 256208 EC50 = 16000 nM T88185 D0FF9F 6485181 EC50 = 85.11 nM T88185 D0G8TM 11483496 EC50 = 48 nM T88185 D0IC7C 776421 EC50 = 109.65 nM T88185 D0J7LY 11436345 EC50 = 240 nM T88185 D0M4BZ 11594881 IC50 = 140 nM T88185 D0M7DC 574310 EC50 = 776.25 nM T88185 D0Q0PN 11494579 IC50 = 13 nM T88185 D0T2KY 44250176 EC50 = 9120.11 nM T88185 D0T2QL 444539 Ki = 4900 nM T88185 D0U6SQ 676464 EC50 = 181.97 nM T88185 D0VE9G 2736690 EC50 = 400 nM T88185 D0W1OR 7424 EC50 > 1000000 nM T88185 D0Y7XK 136127015 IC50 = 370 nM T79694 D0Q4XQ 3291 IC50 > 5000000 nM T79694 D0F4GF 24765479 IC50 = 1.5 nM T79694 D0W8XT 60663 IC50 = 126 nM T79694 D0X5OV 42609962 IC50 = 264 nM T79694 CUQ4R7 2987239 IC50 > 10000 nM T79694 CNZ1F7 6458316 IC50 = 390 nM T79694 CP5NF6 6461757 IC50 = 32 nM T79694 CG8KR9 16005860 IC50 = 32 nM T79694 CJ0C1I 24765309 Ki = 5 nM T79694 C5KA0N 24893979 IC50 = 82 nM T79694 C5AF2Y 25129498 IC50 = 93 nM T79694 C4UC8Q 25129499 IC50 = 7613 nM T79694 CDQ7C1 25129500 IC50 = 552 nM T79694 C0VA5I 25129848 IC50 = 771 nM T79694 CV93JO 25129849 IC50 = 109 nM T79694 CL8YG2 25129850 IC50 = 38 nM T79694 CCB74X 25129851 IC50 = 3480 nM T79694 CJ6TD3 25129852 IC50 = 41 nM T79694 C8PJ6A 25129853 IC50 = 45 nM T79694 C4SA9U 25129854 IC50 = 351 nM T79694 CR08CW 25130208 IC50 = 2552 nM T79694 C10XEL 25130209 IC50 = 1683 nM T79694 C6CB1W 25130210 IC50 = 99 nM T79694 CXK12T 25130211 IC50 = 27 nM T79694 C6CF3U 25130212 IC50 = 97 nM T79694 CS3OY1 25130213 IC50 = 252 nM T79694 CGC5U6 25130214 IC50 = 169 nM T79694 CYD2Q3 25130556 IC50 = 22 nM T79694 CK04RW 25130557 IC50 = 42 nM T79694 C1REU6 35537998 IC50 = 24 nM T79694 COTQ47 44568792 IC50 = 411 nM T79694 CUX2C0 44593418 IC50 = 245 nM T79694 CDC59A 44593419 IC50 = 281 nM T79694 CSD5Z3 44593420 IC50 = 61 nM T79694 CPS12B 53317097 Ki = 1.2 nM T79694 CLXH36 72793718 IC50 = 9000 nM T79694 CLHP58 118560158 IC50 = 2 nM T79694 C9S4YL 118560191 IC50 = 1.8 nM T79694 C0LR9M 118560290 IC50 = 0.92 nM T79694 C7Y8FJ 118560322 IC50 = 1.8 nM T79694 CE6O4V 118560356 IC50 = 3.5 nM T79694 CMAN70 118560393 IC50 = 4 nM T79694 C4VG3F 118560394 IC50 = 1.6 nM T79694 CZ6O0E 118560399 IC50 = 1 nM T79694 CVRO18 118560401 IC50 = 1.1 nM T79694 CZ62GY 118560409 IC50 = 0.89 nM T79694 CL12OZ 118560423 IC50 = 5.4 nM T79694 CH84UX 118560458 IC50 = 1.3 nM T79694 C7Y2LQ 118560466 IC50 = 10 nM T79694 C0JAX6 118560472 IC50 = 3.4 nM T79694 CDJL48 118560488 IC50 = 1.9 nM T79694 CY2KI3 118560543 IC50 = 3.6 nM T79694 C37PDX 118560579 IC50 = 3.3 nM T79694 CG25JS 118560588 IC50 = 2.1 nM T79694 CLK32A 118560592 IC50 = 1.8 nM T79694 C04FRX 118560613 IC50 = 6.1 nM T79694 CB41MH 118560618 IC50 = 7.5 nM T79694 CS0RQ3 118560699 IC50 = 2.6 nM T79694 CQG3K7 118560709 IC50 = 1.8 nM T79694 C2DA9Z 118962193 IC50 = 1.5 nM T79694 CF6D2P 126740597 IC50 = 2.3 nM T79694 CAYS28 126740598 IC50 = 11 nM T79694 CIQ23U 126740608 IC50 = 2.9 nM T79694 C1O5VB 126740610 IC50 = 2 nM T79694 C9KEY6 126740618 IC50 = 4.1 nM T79694 CA1M2Q 126740623 IC50 = 0.76 nM T79694 CNUF36 126740624 IC50 = 1.8 nM T79694 COE64S 126740626 IC50 = 1.7 nM T79694 CS2Y3W 126740650 IC50 = 2.8 nM T79694 CHO17P 126740652 IC50 = 1.2 nM T79694 CKNV98 126740697 IC50 = 6.6 nM T79694 C0AI1V 132991411 IC50 = 11 nM T79694 C1XR9I 134130259 IC50 = 164 nM T79694 C3P7TZ 134130807 IC50 = 14 nM T79694 C9RZB3 134131854 IC50 = 17 nM T79694 CW0Q7I 134132801 IC50 = 25 nM T79694 CHR09A 134133339 IC50 = 133 nM T79694 CG21YN 134133529 IC50 = 259 nM T79694 CE32KO 134133599 IC50 = 33 nM T79694 CH9MI7 134133901 IC50 = 73 nM T79694 C3GIH1 134134030 IC50 = 7 nM T79694 CEWV89 134134318 IC50 = 5 nM T79694 C5RY7Q 134134580 IC50 = 12 nM T79694 CBC5I3 134135133 IC50 = 326 nM T79694 C67QGZ 134135164 IC50 = 4 nM T79694 CV0I4O 134135871 IC50 = 4 nM T79694 CJM8S0 134135899 IC50 = 13 nM T79694 CQ54CZ 134135912 IC50 = 74 nM T79694 CK9MG1 134136380 IC50 = 340 nM T79694 CJ4T0C 134138248 IC50 > 10000 nM T79694 CW4BU5 134138250 IC50 = 20 nM T79694 CLW07U 134138308 IC50 = 9 nM T79694 CERI05 134138759 IC50 = 9 nM T79694 C29IBJ 134139406 IC50 = 148 nM T79694 CPG8R2 134139460 IC50 = 1710 nM T79694 CRJ72V 134140275 IC50 = 4 nM T79694 C9CO2P 134140278 IC50 = 52 nM T79694 C39PGW 134140468 IC50 = 210 nM T79694 C8L5VZ 134140864 IC50 = 5 nM T79694 C62AVQ 134141003 IC50 = 13 nM T79694 C3NRL2 134141387 IC50 = 10 nM T79694 CIPG12 134141754 IC50 = 1000 nM T79694 C90WMC 134141766 IC50 = 100 nM T79694 CR29YW 134141773 IC50 = 15 nM T79694 C4IV9M 134141806 IC50 > 9000 nM T79694 CGA34U 134141893 IC50 = 251 nM T79694 C6U2PJ 134142122 IC50 = 17 nM T79694 C0CT2A 134142164 IC50 = 14 nM T79694 CVC5M6 134142399 IC50 = 306 nM T79694 CXK8D7 134142518 IC50 = 6 nM T79694 C16TWR 134142614 IC50 = 130 nM T79694 C2VSP7 134143155 IC50 = 13 nM T79694 CQ80GN 134143440 IC50 = 8 nM T79694 C1PT9H 134143519 IC50 = 2 nM T79694 CEG7S4 134143554 IC50 = 22 nM T79694 CH03BE 134143575 IC50 = 281 nM T79694 C2VJ7N 134143801 IC50 > 10000 nM T79694 C9A1XL 134143901 IC50 > 8740 nM T79694 CS7G2P 134144179 IC50 = 12 nM T79694 C1OLQ9 134144496 IC50 = 641 nM T79694 C8XR0U 134145066 IC50 = 25 nM T79694 CN8WV9 134145759 IC50 = 8 nM T79694 C6OD8Y 134145781 IC50 = 8 nM T79694 CB6QF0 134145994 IC50 = 10 nM T79694 C7GL6O 134146020 IC50 = 13 nM T79694 CY5ME7 134146171 IC50 = 10 nM T79694 CG7RX1 134146440 IC50 = 308 nM T79694 CN2ST6 134146817 IC50 > 8605 nM T79694 CE15VD 134146997 IC50 = 14 nM T79694 CV73DS 134147142 IC50 = 892 nM T79694 CU0WK1 134147287 IC50 = 243 nM T79694 C1JXF2 134147318 IC50 = 6 nM T79694 C6J0RP 134147643 IC50 = 610 nM T79694 C0ZQM8 134147890 IC50 = 95 nM T79694 C5C7BZ 134147980 IC50 = 139 nM T79694 C9W1AN 134148285 IC50 = 1003 nM T79694 CW9M8G 134148369 IC50 = 12 nM T79694 C45XMS 134148468 IC50 = 6 nM T79694 C20MDR 134148760 IC50 = 46 nM T79694 CWZ47K 134149196 IC50 = 11 nM T79694 C1UY6K 134149672 IC50 = 4 nM T79694 CYQ43A 134149751 IC50 = 473 nM T79694 C4FC6U 134149941 IC50 = 6 nM T79694 CJZ29K 134149992 IC50 > 10000 nM T79694 CML57E 134151608 IC50 = 10 nM T79694 CO1JA4 134151710 IC50 = 95 nM T79694 CV25WH 134151973 IC50 = 97 nM T79694 C0NU4T 134152220 IC50 = 8 nM T79694 CVLO27 134152587 IC50 = 9 nM T79694 C7TV2H 134152703 IC50 = 91 nM T79694 CKI47N 134152745 IC50 = 214 nM T79694 C7NV2W 134152994 IC50 = 23 nM T79694 CFK81J 134153093 IC50 = 1589 nM T79694 C19LMT 134153241 IC50 = 33 nM T79694 CZX13T 134153284 IC50 = 225 nM T79694 CV9ME7 134153508 IC50 = 6 nM T79694 C4L8QS 134153676 IC50 > 10000 nM T79694 C0V6YF 134153738 IC50 = 31 nM T79694 CEA6H8 134153757 IC50 = 137 nM T79694 CMH28S 134154353 IC50 = 3557 nM T79694 C3AW2M 134155076 IC50 = 206 nM T79694 CX8P0D 134155552 IC50 = 26 nM T79694 CN98ZC 134156036 IC50 = 1810 nM T79694 CAS9U3 134156465 IC50 = 55 nM T79694 CE8V5G 134156616 IC50 = 15 nM T79694 C9F3EG 134156994 IC50 = 7 nM T79694 CS4PX9 134157075 IC50 > 10000 nM T79694 C5TC7R 134157194 IC50 = 10 nM T79694 CLMT10 134157774 IC50 = 12 nM T79694 C05KZL 141634203 IC50 = 9 nM T79694 CN9O6Q 145963763 IC50 = 370 nM T79694 CBC6A4 145964052 IC50 = 620 nM T79694 CZFE02 145964073 IC50 = 3.4 nM T79694 C6WB0E 145964120 IC50 = 1370 nM T79694 C1RJ5L 145964213 IC50 = 710 nM T79694 C7TAQ5 145964444 IC50 = 520 nM T79694 CL3J5T 145964488 IC50 > 10000 nM T79694 CX7TC4 145964712 IC50 = 8 nM T79694 C0JGD5 145964736 IC50 > 10000 nM T79694 CUQD06 145964872 IC50 = 1900 nM T79694 C6V5PA 145965039 IC50 = 890 nM T79694 CSJV78 145965046 IC50 = 64 nM T79694 CEK7F5 145965051 IC50 > 10000 nM T79694 CU79FE 145965065 IC50 = 18 nM T79694 C3XZ9G 145965167 IC50 = 6.5 nM T79694 CZ7VP8 145965333 IC50 = 17 nM T79694 COA0D4 145965395 IC50 = 22 nM T79694 CG5D0A 145965520 IC50 > 10000 nM T79694 C2SV8D 145965539 IC50 > 10000 nM T79694 CB24MN 145965576 IC50 = 320 nM T79694 C8MUI9 145965686 IC50 = 810 nM T79694 CM0C4Q 145965785 IC50 = 2250 nM T79694 C74GDJ 145965861 IC50 = 1900 nM T79694 CSR0W9 145965878 IC50 = 6530 nM T79694 CP9GX0 145965960 IC50 > 10000 nM T79694 CC25LD 145966135 IC50 = 9.7 nM T79694 CY6NH0 145966175 IC50 = 2030 nM T79694 C6P5GM 145966272 IC50 = 650 nM T79694 C7MOG0 145966280 IC50 = 420 nM T79694 CNG80S 145966315 IC50 = 2300 nM T79694 C3I5WD 145966882 IC50 > 10000 nM T79694 CB6G2J 145966887 IC50 = 1500 nM T79694 C9OZ7B 145966987 IC50 = 3300 nM T79694 CQ6S4I 145967128 IC50 = 540 nM T79694 CIFN68 145967321 IC50 = 4.7 nM T79694 C3P6KV 145967526 IC50 = 10 nM T79694 CWRS54 145967754 IC50 > 10000 nM T79694 C9GYA8 145968219 IC50 = 1400 nM T79694 C3F9UM 145968918 IC50 > 10000 nM T79694 CO1FC6 145968951 IC50 > 10000 nM T79694 C8A3JX 145968953 IC50 = 7.6 nM T79694 CX2Q3S 145969169 IC50 = 460 nM T79694 C93RXD 145970771 IC50 > 10000 nM T79694 CJE56F 145971412 IC50 = 7.1 nM T79694 CXMQ72 145971782 IC50 = 8600 nM T79694 CM92KQ 145971885 IC50 = 910 nM T79694 CK06VY 145972088 IC50 = 2760 nM T79694 CO0FR7 145972093 IC50 = 1700 nM T79694 CAOS28 145973012 IC50 = 660 nM T79694 C2C1ST 145973030 IC50 = 700 nM T79694 CQYB38 145973089 IC50 = 2.9 nM T79694 C8UN1L 145973107 IC50 = 350 nM T79694 C2L7RP 145973300 IC50 > 10000 nM T79694 CQ7WG9 145973409 IC50 = 380 nM T79694 C1N4UG 145973443 IC50 = 1640 nM T79694 CHZ21U 145973703 IC50 = 2850 nM T79694 CH9P2S 145973704 IC50 = 120 nM T79694 CHQ32U 145973751 IC50 > 10000 nM T79694 C5OX8I 145973789 IC50 = 14 nM T79694 CON93L 145973912 IC50 = 15 nM T79694 CM78OR 145974461 IC50 > 10000 nM T79694 C7B2VG 145974480 IC50 = 1700 nM T79694 C8G1KM 145974485 IC50 = 940 nM T79694 CED15B 145974511 IC50 = 40 nM T79694 C2OL7I 145975061 IC50 = 1150 nM T79694 C9UVC6 145975140 IC50 = 1.6 nM T79694 CDB4P8 145975231 IC50 = 1500 nM T79694 CR2N8T 145975397 IC50 = 5.2 nM T79694 C58WOB 145975751 IC50 = 270 nM T79694 C3W2OE 145975832 IC50 = 4370 nM T79694 C1YSW7 145976102 IC50 = 810 nM T79694 CK8X4G 145976223 IC50 > 10000 nM T79694 CO8KN3 145976268 IC50 > 10000 nM T79694 CN72ZM 145976351 IC50 > 10000 nM T79694 C4KF1L 145976387 IC50 = 980 nM T79694 C3XE5S 145976394 IC50 = 9.8 nM T79694 CE50WI 145976410 IC50 = 2930 nM T79694 CGA1B5 145976660 IC50 = 890 nM T79694 C2BVH9 145976792 IC50 = 7500 nM T79694 C1QU0T 145976799 IC50 = 2360 nM T79694 CM6ZT8 145976855 IC50 = 15 nM T79694 CLCM81 145976857 IC50 = 710 nM T79694 C1L2NM 145977186 IC50 = 67 nM T79694 C0S3TG 145977189 IC50 > 10000 nM T79694 CH3FM6 145977296 IC50 = 40 nM T79694 CAR4F9 145977337 IC50 = 900 nM T79694 C5I6VA 145977340 IC50 = 10 nM T79694 C21VED 145977676 IC50 = 1660 nM T79694 CU38DI 145977733 IC50 = 1800 nM T79694 CSE52C 145977745 IC50 = 1060 nM T79694 C45HOF 145977787 IC50 = 1.8 nM T79694 C1XD8F 145977860 IC50 = 10 nM T79694 CCL06J 145977910 IC50 > 10000 nM T79694 CI89TQ 145978258 IC50 = 110 nM T79694 C8BD3R 145978287 IC50 > 10000 nM T79694 C7DV6A 145978317 IC50 = 7.9 nM T79694 CL36DE 145978466 IC50 = 25 nM T79694 CU0N4O 145978657 IC50 = 2.8 nM T79694 CGW6Q5 145978668 IC50 = 740 nM T79694 D0T6NE 44540045 IC50 = 86 nM T80338 CZN6S9 743974 IC50 > 25118.86 nM T80338 C3VRO9 44557921 IC50 > 10000 nM T80338 C9PAT7 46927672 IC50 = 10 nM T80338 CYX7T2 117072549 IC50 = 7680 nM T80338 C87ZPY 118796358 IC50 > 20000 nM T80338 CEK31P 135566415 IC50 > 20000 nM T80338 CPT0V7 138454752 IC50 = 3130 nM T23714 D04ZBT 6918173 Ki = 0.02512 nM T23714 D05ENJ 11535140 IC50 = 0.05 nM T23714 D0LI1C 44469321 IC50 > 30000 nM T23714 D0X0BI 439201 EC50 = 0.04898 nM T23714 D03ZBM 119343 IC50 = 7 nM T23714 D07OCC 25019714 IC50 = 1.1 nM T23714 D0G0IZ 6918284 Ki = 19 nM T23714 D0ON2X 5311108 IC50 = 1.4 nM T23714 C42UIY 1394282 Ki > 25000 nM T23714 C1P9HQ 9826248 Ki = 21300 nM T23714 C2IQ9X 9830551 Ki = 38 nM T23714 C9SR4E 9874617 IC50 = 0.18 nM T23714 C5RF6H 9894265 IC50 = 2.6 nM T23714 CU15TR 9897921 Ki = 0.1995 nM T23714 CDCM46 9915727 Ki = 69 nM T23714 CK2S7N 9916589 IC50 = 43 nM T23714 CEU3Z2 9916936 Ki = 4 nM T23714 CM45KH 9919335 Ki = 11865 nM T23714 CA54TN 9958759 IC50 = 340 nM T23714 CV6FW9 9987299 Ki = 0.79 nM T23714 CCP49I 9988753 Ki = 1.585 nM T23714 CO4P5L 10005078 Ki = 8900 nM T23714 C0X3IQ 10008626 Ki = 3.981 nM T23714 C4YT1V 10009762 IC50 = 0.26 nM T23714 C7YH1R 10010104 Ki = 0.631 nM T23714 C7JE8F 10010669 Ki = 1.995 nM T23714 CYVZ58 10032884 IC50 = 0.7 nM T23714 CGI57Y 10032895 Ki = 0.631 nM T23714 CNQL86 10055774 Ki = 1.259 nM T23714 CSYU04 10056816 Ki = 2.512 nM T23714 C68GEM 10079793 Ki = 0.631 nM T23714 CIXU90 10079797 Ki = 0.631 nM T23714 CU39IK 10101294 Ki = 0.3981 nM T23714 CF4WK8 10102296 Ki = 0.3981 nM T23714 CXF5K1 10102599 Ki = 0.7943 nM T23714 CY8R9E 10102701 Ki = 0.1259 nM T23714 C4OVQ0 10260476 Ki = 1.585 nM T23714 CHD84V 10327403 Ki = 2.79 nM T23714 C85EUY 10348414 IC50 = 1.1 nM T23714 CJ1W6X 10349694 Ki = 1 nM T23714 CS19JO 10349737 IC50 = 2.4 nM T23714 C8EP5X 10350966 Ki = 0.5012 nM T23714 CR3B4A 10371910 IC50 = 0.51 nM T23714 C8O4XG 10373001 Ki = 770 nM T23714 C1TQ7U 10373970 Ki = 1 nM T23714 CXS0E7 10388673 Ki > 10000 nM T23714 CP14YR 10396101 Ki = 0.3981 nM T23714 CUS3Q8 10418252 Ki = 1 nM T23714 C7X2OY 10418495 Ki = 1.585 nM T23714 CMNA43 10418701 Ki = 0.7943 nM T23714 CXP97A 10439868 Ki = 0.631 nM T23714 C90DQN 10441167 Ki = 0.3981 nM T23714 CX79PI 10441194 Ki = 1.259 nM T23714 C49PQN 10441297 Ki = 0.1995 nM T23714 CJ7CL0 10461651 Ki = 57 nM T23714 C45PFV 10463758 Ki = 0.3981 nM T23714 CWHI15 10463818 Ki = 0.631 nM T23714 C3ZU0G 10463883 Ki = 0.631 nM T23714 CDP56I 10482991 Ki = 46 nM T23714 CN81HS 10506663 IC50 = 610 nM T23714 CNSC12 10507644 IC50 > 10000 nM T23714 C6QBL7 10507708 IC50 = 270 nM T23714 CWJZ47 10508305 IC50 = 180 nM T23714 C67NUL 10530740 IC50 = 130 nM T23714 CWC36F 10531338 IC50 = 160 nM T23714 C8JW7X 10531497 IC50 = 4.6 nM T23714 CM98VJ 10531744 IC50 = 44 nM T23714 C8YX9R 10554743 IC50 = 590 nM T23714 CTRH14 10555061 IC50 = 240 nM T23714 C8NKC1 10555195 IC50 = 39 nM T23714 C5W6HY 10555202 IC50 = 4200 nM T23714 C49EZB 10555263 IC50 = 94 nM T23714 C14JZQ 10555818 IC50 = 3.2 nM T23714 C6E8WS 10556247 IC50 = 11 nM T23714 C93HSP 10556495 Ki = 1430 nM T23714 C73QNP 10578612 IC50 = 8.5 nM T23714 C82NTH 10579143 IC50 = 860 nM T23714 CVE20K 10579159 IC50 = 210 nM T23714 CS3G1W 10579332 IC50 = 3.1 nM T23714 C8V6MZ 10579547 IC50 = 570 nM T23714 C9ZS5F 10579723 IC50 = 510 nM T23714 CC61TV 10580156 IC50 = 7.5 nM T23714 C37LVD 10580536 IC50 = 4.8 nM T23714 C6V9PM 10601892 IC50 = 4100 nM T23714 CEN1B8 10603710 IC50 = 3.9 nM T23714 C6W5CU 10603884 IC50 = 480 nM T23714 CO0L4K 10603982 IC50 = 8400 nM T23714 CJ0Z8R 10604425 IC50 = 150 nM T23714 CZ3I9K 10604560 IC50 = 75 nM T23714 C8H4VG 10604613 IC50 = 4.1 nM T23714 C3R5MZ 10626599 IC50 > 10000 nM T23714 C0X3WA 10626618 IC50 = 110 nM T23714 CQ3H2K 10627129 IC50 = 9100 nM T23714 C3RND6 10627384 IC50 = 0.26 nM T23714 C2I8GS 10627456 IC50 = 350 nM T23714 CJKH95 10627732 IC50 = 14 nM T23714 CC2FB6 10650330 IC50 = 58 nM T23714 C6LE0C 10651068 IC50 > 10000 nM T23714 C8SJ9C 10651074 IC50 = 56 nM T23714 CT1A0W 10651301 IC50 = 150 nM T23714 C5B6LI 10651302 IC50 = 140 nM T23714 C2K3NS 10651897 IC50 = 1.8 nM T23714 C3CK2J 10651980 IC50 = 20 nM T23714 CFZE40 10652092 IC50 = 3.7 nM T23714 CA8C4G 10674242 IC50 = 17 nM T23714 CJGF31 10674687 IC50 = 9.3 nM T23714 C47AXW 10675163 IC50 = 260 nM T23714 C0GP6J 10675204 IC50 = 48 nM T23714 CF43MJ 10675243 IC50 = 4.2 nM T23714 C9ZB5G 10675847 IC50 = 1.6 nM T23714 COD4C2 10698666 IC50 = 150 nM T23714 CVQ3Z9 10698671 IC50 = 1.9 nM T23714 CX36QY 10699094 IC50 = 2000 nM T23714 C62NJO 10699672 IC50 = 16 nM T23714 CX8Q9G 10721082 IC50 = 470 nM T23714 C1TO5J 10721752 IC50 = 7.2 nM T23714 CDG67H 10722378 IC50 > 1000 nM T23714 C3GUO0 10722424 IC50 = 2.2 nM T23714 C9QYO0 10722735 IC50 = 5200 nM T23714 C2CWL8 10734905 Ki > 100000 nM T23714 CGZE45 10744917 IC50 = 150 nM T23714 C95ZHG 10745254 IC50 = 4.8 nM T23714 CE09DK 10745895 IC50 = 79 nM T23714 CT32ZA 10746610 IC50 = 61 nM T23714 C8D7HY 10769383 IC50 = 8.5 nM T23714 CG9EV2 10769485 IC50 = 5.8 nM T23714 CU26PG 10769517 IC50 = 46 nM T23714 CWTM27 10792967 IC50 = 710 nM T23714 CRGJ62 10793125 IC50 = 670 nM T23714 C3J2IM 10793528 IC50 = 670 nM T23714 CQ98CG 10793563 IC50 = 2.5 nM T23714 C1YN4E 10818058 IC50 = 30 nM T23714 CW1S8J 10818426 IC50 = 20 nM T23714 CZL7N4 10840241 IC50 = 3000 nM T23714 CCT9R4 10840498 IC50 > 10000 nM T23714 C71QRE 10840534 IC50 = 830 nM T23714 C2P1DC 10841393 IC50 = 22 nM T23714 CBNE03 10841531 IC50 = 26 nM T23714 CEY5X2 10841582 IC50 = 200 nM T23714 C30WRQ 10841637 IC50 = 1900 nM T23714 CEN18V 10842026 IC50 > 1000 nM T23714 CM5J3S 10842202 IC50 = 2.6 nM T23714 CPI0O9 10876210 Ki = 253 nM T23714 CUJ6H0 11050689 Ki = 237 nM T23714 C1K3VC 11136263 Ki = 1.47 nM T23714 C3D4SJ 11158089 IC50 = 8.1 nM T23714 CQN38W 11158136 IC50 > 1000 nM T23714 CVC71F 11169752 IC50 = 3.5 nM T23714 CYX7C8 11169915 IC50 = 13 nM T23714 CQ2F9B 11169975 IC50 = 1.2 nM T23714 C67ZQB 11180561 Ki > 10000 nM T23714 C7X9MR 11181524 IC50 = 2.5 nM T23714 C49NGS 11193509 IC50 = 2.5 nM T23714 CRF2B9 11204664 IC50 = 1.8 nM T23714 C0A2SL 11204833 IC50 = 1.4 nM T23714 CP0DT6 11215913 Ki = 35000 nM T23714 CB6CK4 11216111 IC50 = 77 nM T23714 CQ04GL 11227059 Ki > 10000 nM T23714 CF8UZ0 11227974 IC50 = 0.43 nM T23714 C7JH4E 11239019 IC50 = 1 nM T23714 CFY6E8 11239502 IC50 = 61 nM T23714 C0KN3B 11239595 IC50 = 0.64 nM T23714 CT59CZ 11250929 IC50 = 34 nM T23714 CWJQ14 11251046 IC50 = 0.47 nM T23714 CUB4Z0 11262728 IC50 = 0.36 nM T23714 CTJW92 11284303 Ki = 1400 nM T23714 CYX1M4 11308648 IC50 = 1.6 nM T23714 CS5EH9 11319515 Ki > 10000 nM T23714 CU4M0J 11320262 IC50 = 2.4 nM T23714 C7IL8N 11342079 Ki = 13300 nM T23714 C8NXI7 11343115 IC50 = 2.6 nM T23714 CJ8LZ5 11365433 Ki > 10000 nM T23714 C79ZES 11411594 IC50 = 0.52 nM T23714 C2FO9H 11411675 IC50 = 0.4 nM T23714 C1A7IM 11422541 IC50 = 0.91 nM T23714 C2XF9D 11422667 IC50 = 5.9 nM T23714 CFE14G 11433973 IC50 = 1.4 nM T23714 CFG04P 11444808 Ki > 10000 nM T23714 C2T0GL 11445066 IC50 = 1.6 nM T23714 CRB59D 11445540 IC50 = 0.69 nM T23714 C6F2IJ 11456652 IC50 = 1.1 nM T23714 C6DGB7 11467345 Ki = 15000 nM T23714 CHK4G3 11468071 IC50 = 2500 nM T23714 C65HWQ 11468276 IC50 = 1 nM T23714 C6AWK4 11479739 IC50 = 0.56 nM T23714 C98PKD 11490605 IC50 = 4.2 nM T23714 CJ37IS 11490839 IC50 = 0.28 nM T23714 CV6S7H 11491041 IC50 = 0.42 nM T23714 CFV1J2 11491055 IC50 = 0.83 nM T23714 CH95EY 11491069 IC50 = 3.7 nM T23714 C4RKM5 11495796 Ki > 10000 nM T23714 C13DVN 11498691 Ki = 398.11 nM T23714 C4BD2X 11498853 Ki = 0.05012 nM T23714 CNT5H8 11505970 Ki = 19.95 nM T23714 C5SPA8 11506007 Ki = 3.981 nM T23714 CO7HB4 11513104 Ki = 7943.28 nM T23714 C5M2QO 11513163 Ki = 100 nM T23714 CVL4R2 11513471 Ki = 10 nM T23714 CV97KH 11527838 Ki = 10 nM T23714 C4QK9A 11527892 Ki = 794.33 nM T23714 CR14MO 11527906 Ki = 7.943 nM T23714 CF37AZ 11542210 Ki = 630.96 nM T23714 CWLX79 11546560 Ki > 10000 nM T23714 C4B8LI 11549335 Ki = 158.49 nM T23714 CMIS36 11549560 Ki = 125.89 nM T23714 CU95QM 11549562 Ki = 158.49 nM T23714 CR5V6E 11553268 Ki > 10000 nM T23714 CUDQ72 11571204 Ki = 316.23 nM T23714 C3ZQ1H 11575578 Ki > 10000 nM T23714 CCF8U0 11577748 Ki = 19.95 nM T23714 C5JY3H 11585604 Ki = 199.53 nM T23714 C7KN1L 11585627 Ki < 10000 nM T23714 CG0Q6N 11589876 Ki > 10000 nM T23714 C7XDG2 11592927 Ki = 39.81 nM T23714 CL9M5H 11600186 Ki = 0.5012 nM T23714 CF5YX0 11600235 Ki = 199.53 nM T23714 C90SJN 11600324 Ki = 0.05012 nM T23714 CW28IT 11604201 Ki > 10000 nM T23714 C1D2NQ 11614670 Ki = 316.23 nM T23714 CXV40U 11620238 Ki > 10000 nM T23714 CRW92U 11621618 Ki = 158.49 nM T23714 C0XZ1G 11621850 Ki = 158.49 nM T23714 CJAD90 11636064 Ki = 398.11 nM T23714 CC0P7Y 11636119 Ki = 79.43 nM T23714 CPR35B 11636121 Ki = 25.12 nM T23714 CL7N1Z 11641218 Ki > 10000 nM T23714 C5PZ3J 11650337 Ki = 63.1 nM T23714 CFB32S 11650783 Ki = 79.43 nM T23714 C9DON1 11657717 Ki = 2511.89 nM T23714 C42RFY 11670114 Ki > 10000 nM T23714 CO5R3C 11671905 Ki = 7943.28 nM T23714 CFA5K1 11672186 Ki = 199.53 nM T23714 C65VUE 11672243 Ki = 199.53 nM T23714 C06SLD 11679144 Ki = 25.12 nM T23714 C5QC8X 11686256 Ki < 10000 nM T23714 C1R7VL 11686399 Ki = 79.43 nM T23714 C8Y4US 11699718 Ki = 100 nM T23714 CZB59C 11707335 Ki = 199.53 nM T23714 C4PY9R 11707423 Ki = 39.81 nM T23714 C4CA1S 11707528 Ki = 251.19 nM T23714 CYG71V 11714620 Ki < 10000 nM T23714 C28ZVE 11719314 Ki > 10000 nM T23714 C8Q6ZV 11757682 Ki > 10000 nM T23714 C3NI6Q 11766718 Ki = 0.1995 nM T23714 C31JUX 11786597 Ki > 10000 nM T23714 CML2Z9 11800992 IC50 = 14 nM T23714 CUP4E3 11801083 IC50 = 130 nM T23714 CM64AW 11801411 IC50 = 730 nM T23714 CN2H5C 11801594 IC50 = 2900 nM T23714 C8UCY2 11801800 IC50 = 14 nM T23714 CX3D7V 11801941 IC50 = 190 nM T23714 CAC92E 11801968 IC50 = 5.2 nM T23714 C19QPM 11802476 IC50 = 1.5 nM T23714 CI98JC 11802489 IC50 = 9.1 nM T23714 CJ24FL 15952860 Ki = 23 nM T23714 C48JMD 16102881 IC50 > 10000 nM T23714 CCHB78 16102882 IC50 > 10000 nM T23714 C6EJP9 16102883 IC50 > 10000 nM T23714 C03DLN 16102884 IC50 > 10000 nM T23714 CAQ93H 16102885 IC50 > 10000 nM T23714 CYN40W 16102907 IC50 > 10000 nM T23714 CXZ5J9 16102908 IC50 > 10000 nM T23714 C68KPL 16102909 IC50 > 10000 nM T23714 CB43PJ 16105690 Ki = 0.1259 nM T23714 CC7S8Z 16105694 Ki = 0.2512 nM T23714 CLM34B 16105696 Ki = 0.1995 nM T23714 CZ8PH5 16105698 Ki = 0.2512 nM T23714 CXK4E7 16105701 Ki = 0.5012 nM T23714 CB4N2X 16105703 Ki = 0.07943 nM T23714 C8U2YI 16105727 Ki = 0.3162 nM T23714 CVI42S 16105729 Ki = 0.631 nM T23714 CICB86 16105734 Ki = 0.1 nM T23714 CR85GM 16105742 Ki = 0.3162 nM T23714 CFQ42K 16105746 Ki = 0.05012 nM T23714 C6LSG9 16105751 Ki = 0.1585 nM T23714 CL7R0B 16108960 Ki = 49200 nM T23714 C12LZJ 16108962 Ki > 20000 nM T23714 CBL7U8 16108965 Ki = 16000 nM T23714 CL90BF 16108967 Ki = 56000 nM T23714 CMX85A 16108969 Ki = 57000 nM T23714 C43YPA 18923274 IC50 = 510 nM T23714 CM9R6I 19603349 IC50 = 2.2 nM T23714 CDN3I5 22288562 Ki = 300 nM T23714 CQ4Z7I 22288574 Ki = 121 nM T23714 CO6NE1 22288578 Ki = 34 nM T23714 CTB28M 22288581 Ki = 38 nM T23714 CXN9M5 22288598 Ki = 204 nM T23714 CEUF74 22288602 Ki = 3890 nM T23714 CK1EH0 44189787 IC50 = 50 nM T23714 C07CFX 44189789 IC50 = 110 nM T23714 CZ92OM 44189790 IC50 = 3600 nM T23714 CX4YF5 44189791 IC50 = 7100 nM T23714 CG0N7O 44189792 IC50 = 135 nM T23714 C0PR4Q 44190077 IC50 = 68 nM T23714 CS1HZ0 44190165 IC50 = 420 nM T23714 CT7QR8 44190166 IC50 = 67 nM T23714 C26CMG 44190167 IC50 = 64 nM T23714 C0LNZ2 44190168 IC50 = 200 nM T23714 C9LJF8 44190169 IC50 > 5000 nM T23714 CYJ7S2 44190263 IC50 = 1.8 nM T23714 C38DGB 44190266 IC50 = 980 nM T23714 CWR0B2 44190267 IC50 = 80 nM T23714 CS95GJ 44190268 IC50 = 210 nM T23714 C7QU2W 44190269 IC50 = 20 nM T23714 CBX1W9 44190361 IC50 = 430 nM T23714 CU86YN 44190363 IC50 = 5300 nM T23714 C6ZJ9E 44190581 IC50 = 3.8 nM T23714 CDN69I 44190672 IC50 = 1600 nM T23714 C3EL2H 44190751 IC50 = 29 nM T23714 CD2T0O 44190752 IC50 = 18 nM T23714 CTNF18 44190753 IC50 = 7.5 nM T23714 C9KQ3X 44190754 IC50 = 37 nM T23714 CZ0B2I 44190755 IC50 = 6.5 nM T23714 C7SF0M 44190756 IC50 = 73 nM T23714 CQUV86 44190850 IC50 = 7.8 nM T23714 CJHU58 44190851 IC50 = 2.8 nM T23714 CV89EH 44190852 IC50 = 8.3 nM T23714 C7NL4B 44190853 IC50 = 190 nM T23714 C1QSR9 44190854 IC50 = 12 nM T23714 CQXD83 44190941 IC50 = 14 nM T23714 CW76PS 44190942 IC50 = 3.6 nM T23714 CDY8I9 44190943 IC50 = 140 nM T23714 C6E8LT 44190944 IC50 = 1.4 nM T23714 CMV52H 44191040 IC50 = 0.54 nM T23714 C4A1FB 44191138 IC50 = 580 nM T23714 C8F9XG 44191220 IC50 = 200 nM T23714 CX5ZK8 44191221 IC50 = 4400 nM T23714 CQ60WJ 44191223 IC50 = 760 nM T23714 CBQX69 44191224 IC50 = 200 nM T23714 CI1K4D 44191225 IC50 = 32 nM T23714 C5AUJ7 44191226 IC50 = 310 nM T23714 CY79RP 44214214 IC50 = 0.23 nM T23714 C4XEF9 44215784 Ki = 271 nM T23714 C8OF6B 44215785 Ki = 103 nM T23714 C98IMC 44276287 Ki = 1790 nM T23714 CGPV36 44276375 Ki = 2370 nM T23714 CTXJ53 44276380 Ki = 239 nM T23714 CN7CV8 44276438 Ki = 126 nM T23714 C52KWQ 44276439 Ki = 304 nM T23714 CQB17X 44276455 Ki = 55 nM T23714 C65QIF 44276459 Ki = 44 nM T23714 C0YX5C 44276460 Ki = 10 nM T23714 C97HVN 44276461 Ki = 141 nM T23714 C3LX2U 44276474 Ki = 304 nM T23714 C0BMI5 44276482 Ki = 27 nM T23714 CZ8K7A 44276487 Ki = 5500 nM T23714 CX8VK2 44276488 Ki = 74 nM T23714 CXC5Y9 44276513 Ki = 29 nM T23714 C32JSE 44276550 Ki = 19 nM T23714 C7LCS2 44276599 Ki = 76 nM T23714 CR74NF 44276624 Ki = 752 nM T23714 CWYP51 44276666 Ki = 476 nM T23714 CN0PD1 44276667 Ki = 92 nM T23714 C7H9AX 44276711 Ki = 2290 nM T23714 CKMF30 44276716 Ki = 514 nM T23714 C1PG2H 44276753 Ki = 1710 nM T23714 C7YWV2 44276793 Ki = 15 nM T23714 CRYX93 44276840 Ki = 73 nM T23714 CREQ14 44276841 Ki = 869 nM T23714 CS4QV0 44298960 Ki = 33 nM T23714 C79MBV 44300140 Ki = 4950 nM T23714 C35MPB 44320168 Ki = 410 nM T23714 CTS5K2 44329173 IC50 = 0.36 nM T23714 C4JM8N 44337425 Ki = 6.3 nM T23714 CZ52BE 44337466 Ki = 27 nM T23714 C1DC9O 44337475 Ki = 0.15 nM T23714 CHJ5D7 44337476 Ki = 6.8 nM T23714 C0JFM3 44337489 Ki = 7.7 nM T23714 C7RL4C 44337490 Ki = 0.57 nM T23714 CRIM26 44346103 Ki = 3300 nM T23714 C2TXN8 44346188 Ki > 25000 nM T23714 CL1UE9 44346281 Ki = 1100 nM T23714 C0MR8U 44346283 Ki = 3400 nM T23714 C38HZG 44346306 Ki = 210 nM T23714 C6SX7G 44346347 Ki = 2540 nM T23714 C47EBP 44346361 Ki = 5300 nM T23714 CAC95P 44346364 Ki > 25000 nM T23714 C90XSM 44346367 Ki = 1300 nM T23714 C6NFP1 44346369 Ki > 25000 nM T23714 C52YEQ 44346389 Ki = 3150 nM T23714 CKS6M8 44346449 Ki = 820 nM T23714 CEF94M 44346451 Ki = 17900 nM T23714 C7IB9L 44346464 Ki = 20700 nM T23714 CW13UE 44346668 Ki > 25000 nM T23714 CT2NU1 44347551 Ki = 10000 nM T23714 COG52H 44347756 Ki = 8000 nM T23714 C2AUV7 44353012 IC50 = 120 nM T23714 CK19AE 44355038 Ki = 13 nM T23714 C6TQ2W 44355196 Ki = 14 nM T23714 CN9HK3 44355233 Ki = 0.7 nM T23714 C7FS1Y 44355234 Ki = 6 nM T23714 C9V5OD 44355241 Ki = 1030 nM T23714 CV13OD 44355256 Ki = 18600 nM T23714 CRGM29 44355257 Ki = 770 nM T23714 C32CEM 44355287 Ki = 520 nM T23714 CNE16L 44355288 Ki = 2070 nM T23714 CUI86M 44355289 Ki = 4900 nM T23714 C2WJ1F 44355427 Ki = 2.5 nM T23714 C2PTE1 44355428 Ki = 0.07 nM T23714 CQ6C3X 44360533 IC50 = 0.41 nM T23714 CHJ1E5 44360553 IC50 = 1.5 nM T23714 C27YRK 44360597 IC50 = 0.37 nM T23714 C5C0BW 44360617 IC50 = 3.9 nM T23714 C4LV8K 44360818 IC50 = 0.52 nM T23714 COE3G8 44360877 IC50 = 0.41 nM T23714 C1Y7QS 44360879 IC50 = 4.6 nM T23714 CKUH60 44360968 IC50 = 0.51 nM T23714 CD7SP1 44361029 IC50 = 3.2 nM T23714 CX7PO6 44361827 Ki > 100000 nM T23714 CUM0A5 44361937 Ki = 9200 nM T23714 C5OFW7 44361938 Ki > 100000 nM T23714 C8E2QR 44410425 Ki = 100 nM T23714 CDR6P7 44410526 Ki = 3162.28 nM T23714 CLI08P 44412007 Ki = 0.3981 nM T23714 C4KJR5 44412412 Ki = 25.12 nM T23714 CNZG76 44418930 IC50 > 10000 nM T23714 C79FXT 44421279 Ki > 10000 nM T23714 C4DL5C 44469677 IC50 > 10000 nM T23714 CZD4C2 45261901 IC50 = 2.5 nM T23714 C0PCR6 45265170 IC50 = 2.8 nM T23714 CU90ND 45266115 Ki = 430 nM T23714 C2JTQ1 45266116 Ki = 60 nM T23714 CGY86R 45266117 Ki > 100000 nM T23714 C6MR4C 45266118 Ki = 2570 nM T23714 CC4O0Y 45266119 Ki = 3250 nM T23714 C0TK1M 45266120 Ki = 140 nM T23714 CAN6K8 45266121 Ki = 70 nM T23714 CYZ62K 45266123 Ki = 1030 nM T23714 C91LGT 45266124 Ki = 3440 nM T23714 CO83HR 45266126 Ki = 2700 nM T23714 CD31RX 45266127 Ki = 7050 nM T23714 C7Q8TF 45266128 Ki = 24900 nM T23714 CQ0AV8 45266129 Ki = 110 nM T23714 CH3L0D 45266130 Ki > 100000 nM T23714 CYMP28 45266131 Ki = 4650 nM T23714 C78AGS 45266250 Ki = 3400 nM T23714 CXYB38 45267862 IC50 = 6 nM T23714 CTW3F1 45269613 IC50 = 0.67 nM T23714 CB25TO 45272156 IC50 = 1.3 nM T23714 CAH64U 46905665 Ki = 3300 nM T23714 C6QB4X 46905666 Ki = 60 nM T23714 C8T1GE 46905667 Ki > 100000 nM T23714 C1JIE9 46905668 Ki > 100000 nM T23714 C7V8CH 46905669 Ki = 1000 nM T23714 CH7JC9 46905670 Ki = 25000 nM T23714 C35IZK 46905894 Ki = 760 nM T23714 CQ4YS6 46905895 Ki = 250 nM T23714 C6Y8JP 46905896 Ki = 800 nM T23714 CZ3XH1 49796348 Ki = 210 nM T23714 CBQ70Z 51351563 Ki = 15800 nM T23714 C7W1CO 57390466 Ki = 0.0631 nM T23714 CUAX92 57391276 Ki = 0.7943 nM T23714 CEI42Q 57391278 Ki = 0.05012 nM T23714 CR4CU9 57392146 Ki = 0.1995 nM T23714 CYDF85 57393059 Ki = 0.631 nM T23714 CAC8M5 57393061 Ki = 0.3162 nM T23714 COG8S6 57394779 Ki = 0.1995 nM T23714 C8PVE2 57394782 Ki = 0.05012 nM T23714 C2TQ5A 57394783 Ki = 0.3981 nM T23714 CJE35F 57396534 Ki = 0.07943 nM T23714 C97VSN 57396535 Ki = 0.2512 nM T23714 C8UG2C 57396537 Ki = 0.1 nM T23714 C5FV8O 57396539 Ki = 0.2512 nM T23714 CK3S0J 57397547 Ki = 0.07943 nM T23714 CM07WZ 57398323 Ki = 0.07943 nM T23714 CG5S2A 57398325 Ki = 0.03981 nM T23714 CDVK40 57398327 Ki = 0.631 nM T23714 CV2NF8 57399227 Ki = 0.07943 nM T23714 C8VG0D 57399981 Ki = 0.0631 nM T23714 C5BK7O 57399982 Ki = 0.2512 nM T23714 C4KTX6 57400985 Ki = 0.1259 nM T23714 C05JCX 57401770 Ki = 0.1 nM T23714 C1JMA0 57401772 Ki = 0.1 nM T23714 C91ALU 57401773 Ki = 0.05012 nM T23714 CJX89L 57401775 Ki = 1 nM T23714 CB0I3M 57401777 Ki = 0.0631 nM T23714 C0HP6R 57401779 Ki = 0.7943 nM T23714 CB4T8H 57401781 Ki = 0.5012 nM T23714 CB2XH5 57401783 Ki = 0.1585 nM T23714 C3C9JU 57402744 Ki = 0.1259 nM T23714 COK10P 57402745 Ki = 0.1259 nM T23714 CG0VE7 57403503 Ki = 0.05012 nM T23714 CT74HP 57403504 Ki = 0.3981 nM T23714 C6Z9WM 70688994 Ki = 43000 nM T23714 C0YZ2D 70695304 Ki = 130 nM T23714 C6B0OV 71450888 Ki = 0.7 nM T23714 CN15EF 71450890 Ki = 160 nM T23714 C5TBC2 71456177 Ki = 140 nM T23714 C9UHA1 71456185 Ki = 11900 nM T23714 CK01OM 71459890 Ki = 162 nM T23714 CWH6T3 72548703 IC50 = 21 nM T23714 C84XQF 73345909 Ki = 7.9 nM T23714 CJ2I4X 73346673 Ki = 0.166 nM T23714 CXR9C8 73346674 Ki = 12.02 nM T23714 C4QLS2 73346675 Ki = 8.913 nM T23714 C3YV0W 73348185 Ki = 0.3981 nM T23714 CE1WK4 73348186 Ki = 2.692 nM T23714 C9MOV6 73348523 Ki = 19 nM T23714 C6WLS1 73349742 Ki = 14.45 nM T23714 CNBL34 73351264 Ki = 0.389 nM T23714 CT72YC 73351265 Ki = 0.2399 nM T23714 CSC0R6 73353239 Ki = 12.59 nM T23714 CO7W1C 73354242 Ki = 575.44 nM T23714 CF49RH 73354498 Ki > 10 nM T23714 CLP8Z0 73354534 IC50 = 0.49 nM T23714 CUK4W3 73355813 Ki = 22.91 nM T23714 CJV89O 73357325 Ki = 0.2042 nM T23714 CWMR48 76331576 Ki = 9.16 nM T23714 C61FVX 90662943 Ki = 62 nM T23714 CSW30M 90662945 Ki = 0.08 nM T23714 CJCV56 90663068 Ki = 44 nM T23714 CKTS63 90663663 IC50 = 3.2 nM T23714 CA0X1D 90663669 IC50 = 2.1 nM T23714 CBZE97 90664274 IC50 = 87 nM T23714 CJM25A 90664281 IC50 = 41 nM T23714 C4W0VE 90664283 IC50 = 98 nM T23714 C5QVG7 90664292 IC50 = 1.1 nM T23714 CFSP80 90664524 IC50 = 19 nM T23714 C49KWZ 90664530 IC50 = 0.28 nM T23714 CBO40Q 90664536 IC50 = 37 nM T23714 CF5UC7 90664542 IC50 = 1.8 nM T23714 CW05GE 90664761 IC50 = 0.76 nM T23714 CM8WH6 90664770 IC50 = 4 nM T23714 CBS98W 90664771 IC50 = 1.2 nM T23714 C6NHL5 90664773 IC50 = 4.8 nM T23714 C1GXB7 90664889 IC50 = 0.88 nM T23714 CY7N1G 90665022 IC50 = 2.7 nM T23714 CZ3A9M 90665033 IC50 = 0.17 nM T23714 CT90YO 90665139 IC50 = 0.26 nM T23714 C6FTK5 90665140 IC50 = 2 nM T23714 CV8O2I 90665141 IC50 = 0.23 nM T23714 C3E1ZP 90665143 IC50 = 0.35 nM T23714 C4J1XG 118719116 Ki = 86 nM T23714 C81PQT 122189902 Ki = 9000 nM T23714 CLR2J7 127034153 IC50 = 20000 nM T23714 C07BQF 10930680 Ki = 34.1 nM T23714 CFTN94 10952583 Ki = 645 nM T23714 CBJ24L 10996140 Ki = 95 nM T23714 CKDA47 11050762 Ki = 119 nM T23714 C3IH6K 44308962 Ki = 299 nM T23714 C2HS8G 44308980 Ki = 4.67 nM T23714 D00FAE 44316621 Ki = 325 nM T23714 D00FUT 123884 Ki > 10 nM T23714 D02DGP 44316161 Ki = 0.4 nM T23714 D04ULY 5312119 Ki = 772 nM T23714 D04WHO 9916412 Ki > 10000 nM T23714 D06QYV 9810391 IC50 = 1.4 nM T23714 D0A3YN 10394861 IC50 = 0.68 nM T23714 D0L3GT 16108961 Ki > 50000 nM T23714 D0LL7N 5311114 IC50 = 0.41 nM T23714 D0N2GM 44316620 Ki = 4.4 nM T23714 D0NY1V 132927 Ki = 60 nM T57613 D06ABF 3957 IC50 = 63400 nM T57613 D02YAQ 6603857 IC50 = 50100 nM T57613 D0J9GD 64715 IC50 = 159000 nM T57613 C7BHW2 60662 IC50 = 24600 nM T57613 CPDW86 252604 IC50 = 23000 nM T57613 CMSU69 738674 IC50 > 30000 nM T57613 CSMB29 759456 IC50 = 150 nM T57613 C5CK1Q 825574 IC50 = 2700 nM T57613 CYX02K 825799 IC50 = 690 nM T57613 CQ62XP 825801 IC50 = 5900 nM T57613 CH30JL 869662 IC50 = 4300 nM T57613 CDM4O2 902575 IC50 = 970 nM T57613 C3FW4S 1019323 IC50 = 710 nM T57613 C16DWN 1085239 IC50 > 30000 nM T57613 C7GE8N 1154076 IC50 = 7100 nM T57613 C2AGB0 1248054 IC50 > 30000 nM T57613 CQ3O0J 1376748 IC50 = 3200 nM T57613 C75PBL 1377831 IC50 = 2200 nM T57613 CEY81D 2840308 IC50 = 1500 nM T57613 C8TSE4 3097786 IC50 > 30000 nM T57613 CMU4F3 3396992 IC50 = 960 nM T57613 C4HMG0 3658964 IC50 = 20000 nM T57613 CH9TO2 3745727 IC50 = 413 nM T57613 CV0W5S 5281899 IC50 = 47700 nM T57613 C95QEX 9540179 IC50 = 2400 nM T57613 CGBE91 9827303 IC50 = 70 nM T57613 CFN1U2 10179495 IC50 = 268100 nM T57613 C9UHG3 11957654 IC50 = 73800 nM T57613 C35GHD 15812076 IC50 > 30000 nM T57613 C57WGP 16219554 IC50 = 45500 nM T57613 C6XP3O 17234805 IC50 = 6500 nM T57613 CFS36C 17234818 IC50 = 2100 nM T57613 C97WQE 17234824 IC50 > 30000 nM T57613 C8A2UI 17234870 IC50 > 30000 nM T57613 CD51EA 17744755 IC50 = 5480 nM T57613 C6RY9W 31520618 IC50 = 330 nM T57613 C2SOY1 46785920 IC50 = 390 nM T57613 CL2A8W 46785922 IC50 = 600 nM T57613 CFZ75O 46880148 IC50 = 480 nM T57613 C0A1CP 49793921 IC50 = 189200 nM T57613 CT2BL8 49842926 IC50 > 30000 nM T57613 CP27XZ 49852186 IC50 > 30000 nM T57613 CLW51Q 49852187 IC50 > 30000 nM T57613 C0NK5Z 49852188 IC50 = 1340 nM T57613 C4UBV9 49852189 IC50 = 2200 nM T57613 CV10JQ 49852190 IC50 > 30000 nM T57613 CL59YO 49852191 IC50 = 12500 nM T57613 C7ZUF5 49852192 IC50 = 5500 nM T57613 CSVZ76 49852193 IC50 = 25000 nM T57613 C6KX1V 49852195 IC50 = 1400 nM T57613 C07TWM 49867945 IC50 = 5600 nM T57613 C5P4AK 49867946 IC50 = 2500 nM T57613 CA2P0D 49867948 IC50 > 30000 nM T57613 CFE80H 49867949 IC50 = 2500 nM T57613 C0Z8FV 49867950 IC50 > 30000 nM T57613 CODR75 50919318 IC50 = 1700 nM T57613 CPF0H1 50919319 IC50 = 38 nM T57613 C13IBD 50919320 IC50 = 750 nM T57613 C1O6QP 51049782 IC50 = 410 nM T57613 CVT26J 51049785 IC50 = 66 nM T57613 C4VQT0 51049787 IC50 = 1000 nM T57613 C7PU3H 51358807 IC50 = 250 nM T57613 C9WS3Z 53301908 IC50 = 730 nM T57613 C9D7AH 53301913 IC50 = 110 nM T57613 C48QEY 53464059 IC50 = 35 nM T57613 CRM42J 58892059 IC50 = 950 nM T57613 C3NS2C 118708433 IC50 = 2300 nM T57613 C3XZY7 118708434 IC50 = 2700 nM T57613 C0AM1J 118708435 IC50 = 2430 nM T57613 D0D3YN 1238 IC50 = 73800 nM T99990 D03ZBT 11626560 IC50 > 10000 nM T99990 D09KTS 24821094 IC50 = 0.5 nM T99990 D0OB0F 5328940 IC50 = 1 nM T99990 D02TUL 118115473 Ki = 545 nM T99990 D03LWG 53235510 IC50 = 3405 nM T99990 D04BFC 59174488 IC50 = 2665 nM T99990 D08AOZ 86582336 IC50 = 32 nM T99990 D0E3TC 44259 IC50 = 6.16 nM T99990 D0G5XV 135565884 IC50 = 0.62 nM T99990 D0H9FR 118295624 IC50 = 272 nM T99990 D0L4FS 5280961 IC50 = 67990 nM T99990 D0QX8X 71479709 IC50 = 37.9 nM T99990 D0YB3W 156414 IC50 = 62 nM T99990 D0T3ME 156422 IC50 > 30000 nM T99990 C9U7NK 1128774 IC50 = 42290 nM T99990 CM5VN6 4600415 IC50 = 38570 nM T99990 CB7WK3 5938113 IC50 = 1900 nM T99990 CUJR40 10062694 EC50 = 30 nM T99990 C0YH2X 11478363 IC50 = 8 nM T99990 CACS26 11561968 Ki > 2000 nM T99990 CU0E8O 11690457 Ki > 10000 nM T99990 C09OWB 16015442 IC50 = 18300 nM T99990 C9TU1O 16046126 IC50 > 1000 nM T99990 C7YG1N 24759534 IC50 = 410 nM T99990 CQNP54 24764449 IC50 = 363 nM T99990 C8B6TY 42628503 EC50 < 500 nM T99990 CEL61X 44229839 IC50 > 10000 nM T99990 CA98KR 44432441 IC50 > 22000 nM T99990 CEQN27 52936621 Ki > 1000 nM T99990 C8ZRE3 53356518 IC50 = 37 nM T99990 C8NA4L 53384644 IC50 > 30000 nM T99990 CJBL48 56925034 IC50 = 119 nM T99990 CE1A9V 57394653 IC50 = 1.53 nM T99990 CV13QY 58540422 IC50 = 14 nM T99990 C1SI3L 59174579 IC50 > 10000 nM T99990 CZ3TG1 59375154 IC50 = 193 nM T99990 CXJ63M 59603829 IC50 = 270 nM T99990 CQEU96 59603842 IC50 = 3.5 nM T99990 CV63UL 67240318 IC50 > 10000 nM T99990 C5DGR9 69036886 IC50 = 1356 nM T99990 C7VJ6A 70647728 IC50 = 24 nM T99990 COU73Y 71226944 IC50 = 20 nM T99990 C40JOZ 71235465 IC50 = 331 nM T99990 CEBO91 71452977 IC50 > 10000 nM T99990 C1SR5V 71576693 IC50 = 7.99 nM T99990 CZ31PU 71583657 IC50 > 10000 nM T99990 C4X1CP 71748056 IC50 = 6.73 nM T99990 CZM1K4 71765510 IC50 = 36 nM T99990 C5MJ0H 71765626 IC50 = 36 nM T99990 CKO8S6 71815907 IC50 = 8.16 nM T99990 C54XWG 72190869 IC50 = 4682 nM T99990 CX75YR 73352604 IC50 = 158.49 nM T99990 CF6QG1 73602845 IC50 = 5.62 nM T99990 CDN83F 73707530 IC50 = 7.36 nM T99990 CCQN01 73775788 IC50 = 15.9 nM T99990 CHF08G 73775789 IC50 = 40.6 nM T99990 COL37D 73775921 IC50 = 18.1 nM T99990 CVQW20 73775923 IC50 = 28.1 nM T99990 C5U4AF 73776059 IC50 = 13.3 nM T99990 CXW54V 73776061 IC50 = 12.9 nM T99990 CD83FL 73776204 IC50 = 19.7 nM T99990 CG84BR 73776205 IC50 = 12.1 nM T99990 C1P3DO 73776206 IC50 = 66.1 nM T99990 CN5D1R 73776207 IC50 = 13.3 nM T99990 CO1C8Y 73776208 IC50 = 8.75 nM T99990 CGC46K 73776360 IC50 = 18.5 nM T99990 C1HW4B 89735655 IC50 = 9800 nM T99990 CAKD54 102594000 IC50 = 83 nM T99990 C8HYU9 117926195 IC50 = 1551 nM T99990 CJGT03 118346182 IC50 = 27.8 nM T99990 C02DGP 118346184 IC50 = 399 nM T99990 CU6NE2 118346192 IC50 = 15.7 nM T99990 CW25VP 118346194 IC50 = 10.5 nM T99990 C37DUM 121293882 IC50 = 13 nM T99990 CXQR89 121294143 IC50 = 3.3 nM T99990 C08KEM 122179540 IC50 = 9700 nM T99990 C3AJ4C 122179546 IC50 > 10000 nM T99990 CG0RP7 122179547 IC50 = 2700 nM T99990 C1A0SQ 122179548 IC50 = 4300 nM T99990 CFKD32 122191637 IC50 = 109 nM T99990 C4X7SD 122192466 IC50 > 10000 nM T99990 CKTJ31 122633242 IC50 > 10000 nM T99990 CUZI17 122633365 IC50 = 2877 nM T99990 C71CNY 122633676 IC50 = 37 nM T99990 C7RXF3 122633687 IC50 = 225 nM T99990 CASW92 122633847 IC50 = 2380 nM T99990 C2ZCK7 122633869 IC50 = 2427 nM T99990 C6UY2L 122633880 EC50 = 197 nM T99990 CQ9MN6 122633890 IC50 = 2562 nM T99990 C5XKI1 122633897 IC50 = 102 nM T99990 CC7P2W 122633900 EC50 = 5.8 nM T99990 CIU72D 127264586 IC50 = 111.2 nM T99990 C0XS4M 129896681 IC50 > 10000 nM T99990 CV89JM 132231876 IC50 = 5.2 nM T99990 C3Z4AT 137321159 IC50 = 3390 nM T99990 C1KSZ6 137475463 IC50 = 1359 nM T99990 C2FT1L 137475480 IC50 = 341.3 nM T99990 CY49JN 137631468 IC50 = 1300 nM T99990 C3X5IR 137631651 IC50 = 3025 nM T99990 C3ME9W 137633853 IC50 = 480 nM T99990 CZOD53 137633880 IC50 = 83 nM T99990 CH50BI 137633922 IC50 = 637 nM T99990 C0SU3Y 137636331 IC50 = 382 nM T99990 C7BJY5 137636807 IC50 = 200 nM T99990 CM27SY 137637237 IC50 > 10000 nM T99990 CU9YQ3 137637635 IC50 = 2420 nM T99990 C03REZ 137638710 IC50 = 591 nM T99990 COS25Z 137638972 IC50 = 4620 nM T99990 C8U1EK 137641775 IC50 > 10000 nM T99990 CFNP52 137642885 IC50 = 4017 nM T99990 CY9S2V 137643114 IC50 = 120 nM T99990 C1RZI5 137643616 IC50 = 1535 nM T99990 CZ89QN 137644872 IC50 = 1263 nM T99990 C6EPW7 137645217 IC50 = 2468 nM T99990 CNUO41 137648000 IC50 = 540 nM T99990 C6BPC3 137648133 IC50 = 2372 nM T99990 CO89DX 137649100 IC50 = 127 nM T99990 C4O9LR 137649355 IC50 = 2823 nM T99990 CN8JP4 137651066 IC50 = 1147 nM T99990 CID46A 137651088 IC50 = 133 nM T99990 C51SDJ 137652231 IC50 = 1544 nM T99990 C1T5MQ 137652396 IC50 = 279 nM T99990 CINE03 137652514 IC50 = 703 nM T99990 C28QUP 137652864 IC50 = 35.7 nM T99990 C31CQF 137654059 IC50 = 86 nM T99990 C32OEN 137654564 IC50 > 10000 nM T99990 CL89XH 137657061 IC50 = 927 nM T99990 C6NPM9 137659694 IC50 = 5160 nM T99990 C23XCP 137661883 EC50 = 18 nM T99990 C57FZP 137662069 IC50 = 33 nM T99990 CPTZ46 137662230 IC50 = 5472 nM T99990 CT02RB 137662268 IC50 = 813 nM T99990 C9ZYG8 141366083 IC50 = 200 nM T99990 C4OD9Q 145967187 IC50 = 174.1 nM T99990 CE31VG 145979714 IC50 = 6310 nM T99990 C9BX4U 145988956 IC50 = 1900 nM T99990 C2MD1Q 155513187 IC50 > 10000 nM T99990 C3NA2I 155519537 IC50 = 83 nM T99990 D01RHR 71519693 IC50 = 1.9 nM T99990 D06BJG 71556703 IC50 = 0.71 nM T99990 D0Q3EW 9549303 IC50 = 386 nM T99990 D0R2WK 16038120 IC50 = 1578 nM T86528 D00NPT 130956 IC50 = 1.9 nM T86528 D08SJZ 60852 Ki = 3.6 nM T86528 D09KLR 2088 Ki = 44.2 nM T86528 D0BF8G 4674 Ki = 55.9 nM T86528 D0PA5S 5245 IC50 = 0.36 nM T86528 D0V8PA 71237 Ki = 63.5 nM T86528 D0VM2L 68740 Ki = 0.07 nM T86528 CPW9G5 65126 IC50 = 20000 nM T86528 CWX8M0 65158 IC50 = 13300 nM T86528 C4GBD1 68686 IC50 > 500000000 nM T86528 CT2Q3V 84770 IC50 = 66650 nM T86528 C9VUZ3 157809 IC50 = 1.288 nM T86528 CC6K8J 165259 Ki = 790 nM T86528 C4TG5Q 169445 IC50 = 30770 nM T86528 CH9E7Z 177788 Ki = 5040 nM T86528 CY2ON3 194564 IC50 > 100000 nM T86528 CD1V5Y 205058 IC50 > 500000000 nM T86528 C0ID4C 405368 Ki = 48.2 nM T86528 C1Q8OH 405370 Ki = 4200 nM T86528 C3ISM5 405374 Ki = 302.6 nM T86528 CNZI26 405380 Ki = 120 nM T86528 CEGR61 405381 Ki = 140 nM T86528 CEI31S 405387 Ki = 1700 nM T86528 C0K5BH 405389 Ki = 23 nM T86528 CEFR19 405390 Ki = 49 nM T86528 CWQS28 405391 IC50 = 18.2 nM T86528 C5I1WQ 405394 Ki = 330 nM T86528 C7O9UK 405400 Ki = 980 nM T86528 CMQ70C 405401 Ki = 47 nM T86528 C3NA8Q 405731 Ki = 41 nM T86528 CR1M0T 406056 Ki = 1500 nM T86528 C5KT6B 406058 Ki = 15 nM T86528 CQEU56 406059 Ki = 180 nM T86528 C25UGC 406061 Ki = 300 nM T86528 CG0MW5 406062 Ki = 7300 nM T86528 C7R8FO 406069 Ki = 3900 nM T86528 C91ECD 406077 Ki = 310 nM T86528 CK6LE9 406400 Ki = 130 nM T86528 CME7Z5 406402 Ki = 40 nM T86528 CXS08P 406404 Ki = 650 nM T86528 C15PZG 406406 Ki = 620 nM T86528 C6MW3U 406408 Ki = 640 nM T86528 CVZ54N 406411 IC50 = 2.692 nM T86528 C0Z1SE 406413 IC50 = 3.917 nM T86528 CTV18L 406415 IC50 = 2.594 nM T86528 CO42GQ 406416 IC50 = 1.047 nM T86528 CVZ85M 413628 IC50 = 1800 nM T86528 CLV4X1 442009 IC50 = 13300 nM T86528 CV2PX1 736818 IC50 > 500000000 nM T86528 CA3UT4 3014316 IC50 > 100000 nM T86528 C2MC5T 4368807 IC50 = 149590 nM T86528 C6V8LU 5238184 IC50 = 1.102 nM T86528 C06USV 5254988 Ki = 10 nM T86528 C34WKT 5276507 Ki = 590 nM T86528 C3CR0F 5276533 Ki = 2.3 nM T86528 CR3EN6 5276543 Ki = 17 nM T86528 CXR17J 5277479 IC50 = 44000 nM T86528 CLNZ13 6451409 Ki = 1880 nM T86528 CX3GZ8 6932064 IC50 > 500000000 nM T86528 CK3P8C 9800268 IC50 = 1.816 nM T86528 C9OEC6 9813652 Ki = 100 nM T86528 CSC61N 9881667 Ki = 400 nM T86528 CR54UA 9903576 IC50 = 17.78 nM T86528 CHA05W 9972123 IC50 = 4.819 nM T86528 CZIV24 10423227 IC50 = 160 nM T86528 CQ02ZF 10424622 Ki = 155.4 nM T86528 CN2E4A 10469336 IC50 = 5.129 nM T86528 CI1YK2 10860031 IC50 = 632.41 nM T86528 C81NQW 10869876 IC50 = 66.68 nM T86528 CZXD64 10883819 IC50 = 246.04 nM T86528 C6VIF2 10927136 IC50 = 18.2 nM T86528 COV26P 10935180 IC50 = 2404.36 nM T86528 C0S1PO 10938511 IC50 = 23.99 nM T86528 CJ7E1W 10946056 IC50 = 50.82 nM T86528 C5W2TN 10949322 IC50 = 10.07 nM T86528 C74WSM 10957079 IC50 = 1.972 nM T86528 CQHO90 10958471 IC50 = 2.692 nM T86528 CBH2Y3 10971795 IC50 = 3.119 nM T86528 CK8A4M 10981675 IC50 = 64.57 nM T86528 CBZV83 11000210 IC50 = 2197.86 nM T86528 CTCJ38 11000619 IC50 = 10.47 nM T86528 CS6T3V 11001596 IC50 = 6.152 nM T86528 CJ8L4Z 11003818 IC50 = 4.266 nM T86528 CJ2ZT0 11011080 IC50 = 18.45 nM T86528 CGP1H0 11011374 Ki = 11.6 nM T86528 CX9VS0 11036766 IC50 = 0.618 nM T86528 C9WMV1 11044348 IC50 = 5.129 nM T86528 CD01AI 11044775 IC50 = 5 nM T86528 C8OX1M 11046047 IC50 = 885.12 nM T86528 CXP8U3 11078699 IC50 = 55.85 nM T86528 CMA39G 11079453 IC50 = 3.89 nM T86528 C89WXY 11080073 IC50 = 3630.78 nM T86528 CRL62I 11080410 IC50 = 1174.9 nM T86528 C4HDL9 11089309 IC50 = 185.35 nM T86528 CDB5C0 11097213 IC50 = 1945.36 nM T86528 CV1BO7 11100705 IC50 = 3.251 nM T86528 CB4MF9 11101324 IC50 = 49.43 nM T86528 C8WP1H 11110387 IC50 = 599.79 nM T86528 C3L0OK 11112420 IC50 = 2.818 nM T86528 CDU5S9 11132684 IC50 = 39.36 nM T86528 C47ABY 11143347 IC50 = 7.079 nM T86528 C0VR4S 11144558 IC50 = 17.99 nM T86528 CW2CS0 11265812 Ki = 900 nM T86528 CA42MY 11336941 IC50 = 470 nM T86528 CL79RT 11728340 IC50 = 3.981 nM T86528 CPED81 11732139 IC50 = 1.445 nM T86528 C3OZ1G 11748130 IC50 = 157.4 nM T86528 CWD4P2 11761251 IC50 = 4.074 nM T86528 C3INL4 11784267 IC50 = 72.11 nM T86528 CI73RU 11784386 IC50 = 1.66 nM T86528 C6Z4AS 11807848 IC50 = 732.82 nM T86528 C31HJW 11811951 IC50 = 17619.76 nM T86528 CL5H1W 11877519 IC50 > 100000 nM T86528 CKUM24 12735335 Ki = 93000 nM T86528 CIJ13G 13855852 IC50 = 18700 nM T86528 CD61CH 13966128 IC50 > 100000 nM T86528 C9EP3Y 15230199 Ki = 3.28 nM T86528 CHR98J 15545194 IC50 = 382 nM T86528 CH5B2T 15602222 IC50 = 7800 nM T86528 CO3P5W 15602227 IC50 = 830 nM T86528 C71VGO 16760285 IC50 = 460 nM T86528 CHB7J8 19069843 Ki = 470 nM T86528 C4L9SZ 19084771 IC50 = 1000000 nM T86528 CDH13A 19084811 IC50 > 10000 nM T86528 CMY15L 19382983 Ki = 310 nM T86528 CZQU17 21219715 IC50 = 3910 nM T86528 CT7ZE3 21745280 Ki = 540 nM T86528 CTA61L 23729568 IC50 > 600000 nM T86528 C6HXL1 23730134 IC50 = 260 nM T86528 CAIZ80 23730138 IC50 = 7943.28 nM T86528 CKV5G7 23730244 IC50 = 27400 nM T86528 CKX32U 23730246 IC50 = 7450 nM T86528 CVC01G 23730248 IC50 = 45600 nM T86528 C5S6DY 23730250 IC50 = 360 nM T86528 C1IMN7 23730362 IC50 = 501.19 nM T86528 CPKV40 23730364 IC50 = 9000 nM T86528 C8I6OE 23730366 IC50 = 1000 nM T86528 CG0K5J 23730367 IC50 = 1000 nM T86528 C0WUS8 23731251 IC50 = 340.4 nM T86528 CHS35C 23731253 IC50 > 600000 nM T86528 CL0BM6 23731254 IC50 > 60000 nM T86528 C3ZUW2 23731256 IC50 = 94.6 nM T86528 CDMP28 25023874 IC50 = 230 nM T86528 CB50SF 25066231 IC50 = 629.5 nM T86528 CG23HZ 44339225 Ki = 16990 nM T86528 C4P7FL 44365667 Ki = 4100 nM T86528 CS50KG 44404469 IC50 = 3570 nM T86528 C86SPQ 44450243 Ki = 128300 nM T86528 C3MHL7 44452344 IC50 > 50000 nM T86528 CR2FG6 44452371 IC50 > 50000 nM T86528 CPVL14 46398840 IC50 = 200 nM T86528 CL6D5C 46398842 IC50 = 80 nM T86528 CIN40U 46886716 IC50 = 10600 nM T86528 C23UTW 46945063 IC50 = 520 nM T86528 C1E2MV 46945064 IC50 = 650 nM T86528 C2OSB3 54669881 IC50 = 150 nM T86528 CBCN04 54673849 IC50 = 430 nM T86528 CX48PZ 54674003 IC50 = 115 nM T86528 C4Q7XW 54674152 IC50 = 164 nM T86528 CS2I0C 54674303 IC50 = 35 nM T86528 CUA6E2 54733930 IC50 > 50000 nM T86528 CXY87D 57384253 IC50 = 115 nM T86528 CIRO63 57384254 IC50 = 47 nM T86528 CI9E6K 57384503 IC50 = 35 nM T86528 C7B3HY 57384508 IC50 = 32 nM T86528 CP7IR9 60198465 IC50 = 310 nM T86528 CL6KO4 70682771 IC50 = 1000 nM T86528 CHT1G0 70687003 IC50 = 12 nM T86528 C52RNJ 70689085 IC50 = 1000 nM T86528 CD18OL 70691191 IC50 = 16 nM T86528 CYMA65 70693295 IC50 > 1000 nM T86528 C4PC9J 70697411 IC50 = 60 nM T86528 C5Q3XG 71521669 IC50 = 57000 nM T86528 CMSO32 71583204 IC50 = 800 nM T86528 CLIB63 71583205 IC50 = 550 nM T86528 CLE62G 71583207 IC50 = 200 nM T86528 CK1Y3W 71583208 IC50 = 22 nM T86528 CI3LB8 71583319 IC50 = 250 nM T86528 C46BWY 71624061 IC50 = 40 nM T86528 CQP0M1 71624063 IC50 = 36 nM T86528 CZO9F3 71624065 IC50 = 80 nM T86528 C15CNH 71624067 IC50 = 230 nM T86528 CFPD04 71624069 IC50 = 320 nM T86528 C4OCQ1 71624071 IC50 = 400 nM T86528 C9UD7T 71624183 IC50 = 2700 nM T86528 CGAP15 71624185 IC50 = 3200 nM T86528 C9R3SV 71624187 IC50 = 7100 nM T86528 C9HQ0L 71624189 IC50 = 170 nM T86528 C4DW8X 71624191 IC50 = 140 nM T86528 CY39BQ 71624193 IC50 = 79 nM T86528 C0X1IZ 71624195 IC50 = 110 nM T86528 CF10RN 71624197 IC50 = 58 nM T86528 CQ9G2H 71624307 IC50 = 44 nM T86528 C81DWJ 71624309 IC50 = 40 nM T86528 CL5H2G 71624311 IC50 = 43 nM T86528 CD0IH6 71624313 IC50 = 110 nM T86528 CB2OI3 71624315 IC50 = 140 nM T86528 C54TJP 71624317 IC50 = 350 nM T86528 C5LBE1 71624436 IC50 = 1100 nM T86528 C4M7IT 71624438 IC50 = 4500 nM T86528 CFBD80 71625848 IC50 = 150 nM T86528 C8DE1G 71625849 IC50 = 49 nM T86528 CHIP97 71625851 IC50 = 34 nM T86528 CBD43U 71625853 IC50 = 30 nM T86528 C40ALH 71625854 IC50 = 49 nM T86528 C5D7AE 71625856 IC50 = 44 nM T86528 C6DU4H 71718590 IC50 = 79000 nM T86528 CZTN60 71720142 IC50 = 140 nM T86528 C78HLF 72376503 IC50 = 39 nM T86528 CKF40R 72712585 IC50 = 21 nM T86528 CXI5E3 72712587 IC50 = 15 nM T86528 CZ9YG4 72712787 IC50 = 200 nM T86528 CK0Q8P 72712788 IC50 = 14 nM T86528 CPWN53 72712789 IC50 = 11 nM T86528 C01ZOP 73351357 IC50 = 84000 nM T86528 C28KJU 74766013 IC50 = 5000 nM T86528 CQF23W 76070739 IC50 = 3300 nM T86528 C52OTJ 76070740 IC50 = 4800 nM T86528 C1VQ7J 76070742 IC50 > 20000 nM T86528 C2M3NU 77108489 IC50 = 28000 nM T86528 C8GFL2 90178625 IC50 = 1200 nM T86528 CY07VO 90185749 IC50 = 1000 nM T86528 CI64RQ 90185765 IC50 = 1500 nM T86528 CRC3A5 90185767 IC50 = 4000 nM T86528 C2H9PS 90645507 IC50 > 20000 nM T86528 C91OBI 90645508 IC50 = 26000 nM T86528 CP9LX7 90656272 IC50 = 33000 nM T86528 C07IKQ 90656274 IC50 = 47000 nM T86528 CB89NF 118732275 IC50 = 1100 nM T86528 CW6ET4 118735930 IC50 = 2000000 nM T86528 CA53FX 118735931 IC50 > 2000000 nM T86528 C4HN0W 124220686 IC50 = 2800 nM T86528 CC3A6Z 124220687 IC50 = 540 nM T86528 C5G3OX 124220688 IC50 >= 100000 nM T86528 CB4S8K 124220689 IC50 = 3700 nM T86528 CWC1L3 127029867 IC50 = 13000 nM T86528 CS69VR 127034117 IC50 = 6600 nM T86528 C3UDB6 132961505 IC50 > 100000 nM T86528 CUP73R 132961507 IC50 = 33300 nM T86528 C7FJ8E 134812642 IC50 > 1000 nM T86528 CWJG84 135262452 IC50 = 2600 nM T86528 C5MF1O 135262453 IC50 = 1000 nM T86528 C3RAT6 135262739 IC50 = 1300 nM T86528 C8B4XY 137633427 IC50 = 8800 nM T86528 CH3T7B 137633467 IC50 = 4600 nM T86528 CVCU81 137634641 IC50 = 1500 nM T86528 CMB92W 137635267 IC50 >= 100000 nM T86528 C9W7PG 137635707 IC50 = 860 nM T86528 CF9L6M 137639739 IC50 = 870 nM T86528 CMP56N 137640726 IC50 = 3000 nM T86528 CCSV43 137640961 IC50 = 1400 nM T86528 C4K0CB 137641721 IC50 = 1100 nM T86528 C04EHY 137643892 IC50 = 2300 nM T86528 CVP74B 137643984 IC50 = 8400 nM T86528 CDXU98 137646839 IC50 = 1000 nM T86528 CLHD09 137647692 IC50 = 2800 nM T86528 CU6NJ2 137649183 IC50 > 100000 nM T86528 C0S8DL 137651980 IC50 = 2600 nM T86528 CX41HG 137653012 IC50 = 4600 nM T86528 CPR6Y0 137654785 IC50 = 1600 nM T86528 C8YP3D 137654832 IC50 = 29800 nM T86528 CQ5H7R 137660616 IC50 = 10000 nM T86528 C4SV5D 137660984 IC50 = 1600 nM T86528 C3F5WZ 139592509 IC50 = 1100 nM T86528 CZ8WT3 139592518 IC50 = 3700 nM T86528 CE8H4R 142463310 IC50 = 62200 nM T86528 CDU34E 142463315 IC50 = 43100 nM T86528 CP1QI3 142463324 IC50 = 71400 nM T86528 CP2B7D 142463326 IC50 > 100000 nM T86528 CF3RI2 142463329 IC50 = 59600 nM T86528 C0LUQ2 145975200 IC50 = 94300 nM T86528 C1LNO5 145982143 IC50 = 41000 nM T86528 C39RYO 145992550 IC50 = 310 nM T86528 CZ65XH 153290116 IC50 = 1400 nM T86528 CZ6E1N 153290133 IC50 = 3000 nM T86528 C9U6WB 155510599 IC50 = 100000 nM T86528 CM65LB 155511026 IC50 > 50000 nM T86528 C2ZJ7D 155511438 IC50 = 2700 nM T86528 CO1FP9 155511573 IC50 = 8000 nM T86528 CVU79A 155512943 IC50 > 100000 nM T86528 CHE5F9 155514899 IC50 = 234 nM T86528 C48UMO 155515171 IC50 = 28000 nM T86528 C7Y6BN 155518110 IC50 = 13300 nM T86528 CQT4F9 155518823 IC50 = 800 nM T86528 CY9TM4 155518943 IC50 = 390 nM T86528 CCRV79 155519974 IC50 = 6030 nM T86528 C7VXC5 155521642 IC50 > 50000 nM T86528 C50PMC 155521922 IC50 > 100000 nM T86528 CP2FJ3 155523119 IC50 = 12500 nM T86528 CMD57U 155523182 IC50 = 41200 nM T86528 C2U9DW 155523692 IC50 = 91200 nM T86528 CIMR81 155524829 IC50 = 2000 nM T86528 C5RNL0 155525423 IC50 = 473 nM T86528 CY1G7P 155526409 IC50 = 150 nM T86528 CW6D4L 155528021 IC50 > 100000 nM T86528 C2S6NJ 155532075 IC50 = 520 nM T86528 CPFQ61 155532616 IC50 = 8100 nM T86528 C4O5PS 155532943 IC50 = 1200 nM T86528 CZ86MI 155533989 IC50 = 252 nM T86528 C2WI7U 155534228 IC50 = 8000 nM T86528 C7XEQ9 155534692 IC50 = 1300 nM T86528 CEX26K 155535100 IC50 = 2700 nM T86528 CL9A3U 155535497 IC50 = 230 nM T86528 C2PB4I 155535609 IC50 = 650 nM T86528 CG0O8S 155536591 IC50 > 100000 nM T86528 CNJ0R4 155538427 IC50 = 81400 nM T86528 C2UKA9 155539163 IC50 = 644 nM T86528 CYUM28 155539260 IC50 > 100000 nM T86528 CZ2DM3 155539327 IC50 > 100000 nM T86528 CICA08 155539437 IC50 > 50000 nM T86528 CW92XV 155539703 IC50 = 1500 nM T86528 CF5Y9N 155541498 IC50 > 100000 nM T86528 CV80JB 155541710 IC50 = 289 nM T86528 C9U0TX 155541923 IC50 = 20000 nM T86528 C9FES8 155542101 IC50 = 35000 nM T86528 COL80H 155542771 IC50 > 100000 nM T86528 CO7TF4 155544562 IC50 = 8600 nM T86528 C5PDE2 155545691 IC50 = 690 nM T86528 CNB36V 155546213 IC50 = 22700 nM T86528 CHUB94 155546327 IC50 = 12500 nM T86528 C2GLV6 155546879 IC50 = 1200 nM T86528 C69ETB 155549431 IC50 = 1100 nM T86528 C4I3EU 155550418 IC50 = 1000 nM T86528 C8JZ0E 155552286 IC50 = 520 nM T86528 CNM1B7 155552416 IC50 = 13700 nM T86528 C5O6JN 155552492 IC50 = 190 nM T86528 CM45VQ 155555314 IC50 = 389 nM T86528 CVS5D9 155556226 IC50 = 2200 nM T86528 CFK5H6 155557012 IC50 = 56300 nM T86528 CM09FD 155560088 IC50 > 100000 nM T86528 CR0O7U 155561075 IC50 > 10000 nM T86528 C0UFQ3 155561537 IC50 = 7400 nM T86528 C3AG7K 155563682 IC50 = 3100 nM T86528 C68HPL 155564810 IC50 = 3000 nM T86528 CDSK47 155565996 IC50 = 25100 nM T86528 CI25BR 155566374 IC50 = 700 nM T86528 CF6H9N 155567024 IC50 = 335 nM T86528 CA1FH7 155568571 IC50 = 1000 nM T86528 D00TEI 54674305 IC50 = 28 nM T86528 D02CYZ 23043575 IC50 = 3069 nM T86528 D02QWB 23043560 IC50 = 9.03 nM T86528 D02SNU 5276531 Ki = 1.09 nM T86528 D03ZDC 9994754 Ki = 3.4 nM T86528 D04TIS 4395717 Ki = 740 nM T86528 D05ONZ 12066684 IC50 = 16.4 nM T86528 D05XLD 57637 Ki = 4.45 nM T86528 D05YIK 5276520 Ki = 240 nM T86528 D06III 10014835 Ki = 61000 nM T86528 D09USO 5277466 IC50 = 8500 nM T86528 D0A4MM 9847474 Ki = 3.9 nM T86528 D0B0LU 25140170 IC50 = 28.1 nM T86528 D0C9LF 25023868 IC50 = 550000 nM T86528 D0DC3N 11606263 IC50 > 10000 nM T86528 D0E4DR 25140171 IC50 = 388.2 nM T86528 D0H4MO 14231197 Ki = 1.6 nM T86528 D0I6YD 5276503 Ki = 230 nM T86528 D0L8QX 128523 Ki = 78 nM T86528 D0MY0R 25140321 IC50 = 883.1 nM T86528 D0N0JL 1023 Ki = 29800 nM T86528 D0P2BY 5277505 IC50 = 16.1 nM T86528 D0R0UV 23730136 IC50 = 240 nM T86528 D0W0FX 406401 Ki = 2.3 nM T86528 D0X1FT 25014899 IC50 = 100 nM T86528 D0Y3XR 10468166 Ki = 7.4 nM T86528 D0Z8EU 405372 Ki = 0.74 nM T83198 D09MSN 74229666 Ki <= 77000 nM T83198 C7H2TY 123137 IC50 > 1000000 nM T83198 CHCF90 665797 EC50 = 13700 nM T83198 COY71L 1073725 Ki = 250 nM T83198 CL5R9D 1733244 Ki = 280000 nM T83198 CI5C4F 2133805 EC50 <= 50000 nM T83198 CF47SL 6420114 Ki = 540 nM T83198 CXP4D9 6875758 EC50 = 9800 nM T83198 CRKZ07 11839291 EC50 <= 25000 nM T83198 C3EW7A 50744391 Ki = 2800 nM T83198 C7PZ9N 56840728 Ki = 560 nM T83198 CM4K7G 70680427 EC50 <= 800000 nM T83198 CX3Q7K 71618700 Ki <= 800000 nM T83198 CAN4Z5 72771091 IC50 = 7400 nM T83198 CP7H8X 72771092 IC50 = 750 nM T83198 C4O1IR 73330369 Ki = 6.1 nM T83198 C8YL5N 73355065 IC50 = 33 nM T83198 C7E1UW 76333050 EC50 = 395 nM T83198 CH9R1G 77461035 IC50 = 110 nM T83198 CBR20Z 91885637 IC50 = 44 nM T83198 C5JVR4 91971266 Ki = 48 nM T83198 CYG4Q3 118169882 IC50 = 47 nM T83198 CVX89N 118169940 IC50 = 24 nM T83198 CVT45P 118170010 IC50 = 42 nM T83198 CGP2N1 118170044 IC50 = 69 nM T83198 CW50PX 118170336 IC50 = 140000 nM T83198 C1KYL6 118170387 IC50 = 10 nM T83198 CMW6L4 118170433 IC50 = 180 nM T83198 C8R1EV 118170437 IC50 = 130 nM T83198 C3PN4G 118170474 IC50 = 3400 nM T83198 C6R4GP 118170531 IC50 = 320 nM T83198 C75ITU 118170752 IC50 = 580 nM T83198 CXD39Z 118170767 Ki = 1 nM T83198 C6KN0M 118170851 IC50 = 2400 nM T83198 CAE2Z4 118170891 IC50 = 270 nM T83198 CLN34U 118188783 IC50 = 37 nM T83198 CYFC56 118952707 IC50 = 700 nM T83198 CER0B2 118952731 IC50 = 100 nM T83198 CVZ8W3 118952733 IC50 = 400 nM T83198 CO6WB4 118952741 IC50 = 200 nM T83198 CS03TX 118952751 IC50 = 200 nM T83198 C1ZE6C 118952781 IC50 = 5400 nM T83198 CA8WJ1 118987021 IC50 = 47000 nM T83198 CQA37M 122180503 Ki <= 800000 nM T83198 COC0V8 122190591 Ki <= 100000 nM T83198 C9G2JO 122194678 IC50 = 2300 nM T83198 CE45IP 122194684 IC50 > 250000 nM T83198 C4KPW8 122194810 IC50 = 400 nM T83198 C7U6SV 122653346 IC50 = 20 nM T83198 CP1SA8 122653376 IC50 = 260 nM T83198 C34IPT 127053094 IC50 = 61000 nM T83198 CJ2OP1 134131661 IC50 = 248 nM T83198 CGP6H4 134141818 IC50 = 115 nM T83198 C3L8XK 134143193 IC50 = 9.45 nM T83198 C9LM1F 134150222 IC50 = 5390 nM T83198 CYQ4O8 134151181 IC50 = 42.6 nM T83198 C4VZ1I 134152048 IC50 = 3570 nM T83198 C0N6YO 134154488 IC50 = 730 nM T83198 CQ3E4F 134156566 IC50 = 29.6 nM T83198 CIE0X2 137637791 IC50 = 290 nM T83198 C62ABF 137638786 IC50 = 260 nM T83198 CS0UX9 137647262 IC50 = 160 nM T83198 C2RDZ7 137650952 Ki = 2.1 nM T83198 C84URZ 137652956 IC50 = 180 nM T83198 CVF24T 137659055 IC50 = 170 nM T83198 C2Z4TL 137797043 IC50 = 170000 nM T83198 C7K4XY 138911332 IC50 = 43 nM T83198 CP0VZ2 139030534 Ki = 13 nM T83198 CTOY58 145949553 IC50 = 20800 nM T83198 C2C3AZ 145950199 IC50 = 63.15 nM T83198 C23HBE 145953152 Ki <= 99000 nM T83198 CE9CB2 145955302 IC50 = 18.31 nM T83198 CTXK74 145955909 IC50 = 8000 nM T83198 CJ62PI 145955936 IC50 = 750 nM T83198 C05EDZ 145958249 IC50 = 69700 nM T83198 CKV9M4 145958345 IC50 = 2200 nM T83198 CN2T3X 145960115 IC50 = 1200 nM T83198 C5OL0F 145975241 IC50 = 10 nM T83198 CX92YA 145982583 Ki = 274.9 nM T83198 CZ7L1C 145984438 Ki = 61.9 nM T83198 C8LFQ9 145984561 Ki = 47.9 nM T83198 C5LG3W 145984572 Ki = 6.1 nM T83198 C9ZV5T 145985825 Ki = 95 nM T83198 C91CJM 145986114 Ki = 151500 nM T83198 C03SXH 145986134 Ki = 47.7 nM T83198 COL28A 146819721 EC50 = 8 nM T83198 C0RL6M 149484089 EC50 = 7 nM T83198 CS2KY6 149845604 EC50 = 33 nM T83198 CMIX17 150024611 EC50 = 24 nM T83198 CSG04X 150380309 EC50 = 45 nM T83198 C1CH5M 151456260 EC50 = 70 nM T83198 CI2W6Q 151590841 EC50 = 6 nM T83198 CVP5F9 151996422 EC50 = 2 nM T83198 C46HNQ 152074111 EC50 = 56 nM T83198 C2H9RZ 154584187 Ki = 50 nM T83198 C8ERJ2 155513129 IC50 = 13760 nM T83198 CK12AF 155513191 IC50 = 550 nM T83198 C0VOE8 155513585 IC50 = 10100 nM T83198 CW3GB0 155514454 IC50 = 30.7 nM T83198 C8HWX1 155514912 IC50 = 300 nM T83198 CS7NF5 155515078 IC50 = 1300 nM T83198 CX5WC9 155516485 IC50 > 1000000 nM T83198 CD08VW 155518083 IC50 = 1490 nM T83198 C51GIZ 155518657 EC50 = 2 nM T83198 CZ29WB 155518662 IC50 = 12370 nM T83198 CNK64L 155521091 IC50 = 7260 nM T83198 C6BMH5 155524211 IC50 = 33280 nM T83198 CKDO19 155524700 IC50 > 50000 nM T83198 CS90HX 155525643 IC50 = 1320 nM T83198 C3YM4N 155526141 IC50 > 50000 nM T83198 C0R5GF 155528221 IC50 = 330000 nM T83198 CSG27X 155528223 IC50 = 18400 nM T83198 CB2S5P 155528969 IC50 = 590 nM T83198 C8KCA6 155529264 IC50 > 50000 nM T83198 CW8M7Y 155529372 EC50 = 18 nM T83198 C3H6MV 155531206 IC50 > 50000 nM T83198 CKI6D1 155531475 IC50 = 11010 nM T83198 C2YSZ6 155533694 IC50 > 50000 nM T83198 C23RQY 155534766 IC50 > 50000 nM T83198 CGD98U 155535168 IC50 = 7010 nM T83198 CBA50J 155536779 IC50 = 15920 nM T83198 CRKA06 155538158 EC50 = 14.7 nM T83198 C5J4WI 155539280 IC50 > 50000 nM T83198 CG5DI9 155539935 IC50 = 4250 nM T83198 C7Z5OQ 155540103 IC50 = 31 nM T83198 CKHN45 155541334 IC50 = 14790 nM T83198 C9ZX0Q 155543066 IC50 = 450 nM T83198 CI2D6N 155544337 IC50 = 4280 nM T83198 CRO97Y 155545851 IC50 = 27740 nM T83198 CA16VE 155547540 IC50 = 1060 nM T83198 CF9U7D 155553582 IC50 = 74 nM T83198 CA56JR 155554374 IC50 > 50000 nM T83198 CA2Z1M 155556167 IC50 = 44000 nM T83198 CPSQ45 155558701 IC50 > 50000 nM T83198 C4L6YB 155558952 IC50 > 50000 nM T83198 CRO8I7 155559884 IC50 = 1590 nM T83198 CUNS23 155563149 IC50 = 33900 nM T83198 C8XES9 155564335 IC50 = 3290 nM T83198 CFJD02 155566325 EC50 = 14 nM T83198 CR3U1F 155566727 IC50 = 2770 nM T83198 CK6U1Q 155568141 IC50 = 1130 nM T83198 CQTZ49 155568159 IC50 = 260000 nM T42000 D0F9FA 5311139 IC50 = 2000 nM T42000 CT7O6B 21580417 IC50 = 4400 nM T42000 C94VLS 57391090 IC50 = 2700 nM T42000 C0P3NW 57398141 IC50 = 15500 nM T42000 CAC6O8 57398142 IC50 = 3700 nM T42000 C5RO1T 57398143 IC50 = 34300 nM T42000 CH41NQ 57401571 IC50 = 37800 nM T42000 CS2UQ8 155535525 IC50 = 7800 nM T76497 D05TPI 72276 IC50 > 1000000 nM T76497 D0U2BH 65064 IC50 = 720 nM T76497 CTK25Q 72277 IC50 > 1000000 nM T76497 CL5SA1 73160 IC50 > 1000000 nM T76497 CNIW58 107905 IC50 = 210 nM T76497 CDZ65K 199472 IC50 = 1450 nM T76497 C8DL9U 449303 Ki = 10 nM T76497 CQK73W 9882981 IC50 > 1000000 nM T76497 CW31OL 11174492 Ki = 80 nM T76497 C2W9KM 11242708 Ki = 35 nM T76497 CF6S2U 11253838 Ki = 588000 nM T76497 C9C8EK 11369021 Ki = 198000 nM T76497 C7GRO6 11426662 Ki = 40000 nM T76497 CKD9L3 11458565 Ki = 1520 nM T76497 CT28PN 11786932 Ki = 109000 nM T76497 C4E0NA 46905386 Ki = 4400 nM T76497 C2YH8E 46905387 Ki = 3500 nM T76497 D0C4VG 449304 Ki = 130 nM T76497 D0RB1V 6419835 IC50 = 1280 nM T78019 D05EAM 4735 IC50 = 300 nM T78019 D0U7OU 3220 IC50 = 3500 nM T78019 CX4WT9 807542 IC50 = 37800 nM T78019 CT5E7N 897520 IC50 = 28100 nM T78019 CR8ME3 1005314 IC50 = 15400 nM T78019 CPQ3D4 1202786 IC50 = 13300 nM T78019 C6W2BG 1241137 IC50 = 9500 nM T78019 C3VIK9 1398345 IC50 = 43800 nM T78019 CVK03C 1515366 IC50 = 44700 nM T78019 C0QUS5 1618640 IC50 = 11000 nM T78019 CE3S9R 1820399 IC50 > 50000 nM T78019 C6ZC3T 2065247 IC50 = 41700 nM T78019 COGK92 2065762 IC50 = 27600 nM T78019 C54MEA 2271133 IC50 = 2400 nM T78019 C9C0OM 2714312 IC50 = 31400 nM T78019 CV9ZH6 2941126 IC50 = 57000 nM T78019 C3UAV2 5791145 IC50 = 48700 nM T78019 CPL6Y5 5869479 IC50 = 1600 nM T78019 CIO71H 5920585 IC50 = 27700 nM T78019 CT39PY 7027182 IC50 = 3000 nM T78019 C85XHT 7509342 IC50 = 69400 nM T78019 CYOS08 8119828 IC50 = 47800 nM T78019 CD6KQ0 11983303 IC50 = 900 nM T78019 C3NIY8 16456878 IC50 = 102000 nM T78019 CGS1V6 17573525 IC50 = 40300 nM T78019 CAL45Z 17600651 IC50 > 100000 nM T78019 CWU92E 20866464 IC50 > 50000 nM T78019 CJKO23 20866499 IC50 > 50000 nM T78019 CU43TM 44395081 IC50 = 1700 nM T78019 CDL04Q 44411559 IC50 = 900 nM T78019 CLS3I6 44411721 IC50 = 2000 nM T78019 CYD6U4 44411824 IC50 = 3100 nM T78019 CJ3F0S 44411825 IC50 = 1900 nM T78019 C1WLY8 44411827 IC50 = 1700 nM T78019 CT79KF 44411937 IC50 = 3700 nM T78019 C62AMZ 44411939 IC50 = 1200 nM T78019 CBXR07 45840460 IC50 = 167100 nM T78019 CEL91T 56923561 IC50 = 109200 nM T78019 C1AQP8 71552278 IC50 = 800 nM T78019 C2IT1Z 91383855 IC50 = 128 nM T78019 CU3RP8 124141953 IC50 = 35 nM T78019 CW36PU 135500982 IC50 = 41500 nM T78019 C0TE5S 135651612 IC50 = 33200 nM T78019 C82HCM 139193964 IC50 = 30 nM T78019 C5FN6E 155532329 IC50 = 15400 nM T67849 D09XZB 123631 IC50 > 50000 nM T67849 D0B3HD 2519 IC50 = 75000 nM T67849 D0E6XR 3062316 IC50 = 30000 nM T67849 D0F8RA 2153 IC50 = 75000 nM T67849 D0J5VR 11625818 IC50 = 1.2 nM T67849 D0R0MW 5329102 IC50 = 12000 nM T67849 D0RU0O 50905713 IC50 < 0.5 nM T67849 D0S5LD 135565596 IC50 < 0.7 nM T67849 D0W5HK 216239 IC50 > 50000 nM T67849 D00UZR 5330286 IC50 > 10000 nM T67849 D01PGR 16123056 IC50 = 43 nM T67849 D01QSO 16654980 IC50 = 110 nM T67849 D03BHZ 52913813 IC50 = 12 nM T67849 D03EZE 25167777 IC50 = 2.5 nM T67849 D03FOP 68947304 IC50 = 10.9 nM T67849 D03IJO 11618268 IC50 = 12.7 nM T67849 D03KAC 1893730 IC50 = 36 nM T67849 D03LWG 53235510 IC50 > 9000 nM T67849 D03XAQ 49784945 IC50 = 500 nM T67849 D06GUA 49784002 Ki = 0.1259 nM T67849 D07EHV 44814409 IC50 > 9100 nM T67849 D07HPJ 11476171 IC50 > 9100 nM T67849 D08QGT 17755052 IC50 = 3 nM T67849 D0C3ZR 10427712 IC50 = 235 nM T67849 D0D8JB 44516953 IC50 = 6 nM T67849 D0I3LO 91933883 IC50 = 23 nM T67849 D0LG7X 86291103 IC50 = 24.5 nM T67849 D0O1LD 11647372 IC50 = 3 nM T67849 D0O6VZ 25254071 IC50 = 6.7 nM T67849 D0O8SJ 72950888 IC50 = 6.2 nM T67849 D0TU7B 58507717 IC50 = 451 nM T67849 D0U3DP 46912230 IC50 = 37 nM T67849 D0UP1Z 51001932 Ki = 0.12 nM T67849 D0VG0D 11977753 IC50 = 5 nM T67849 D0W7HE 56649450 IC50 = 290 nM T67849 D0XD4I 118502708 IC50 = 270 nM T67849 D0Y2NS 70798655 IC50 = 13900 nM T67849 D03BNU 59604787 IC50 > 5000 nM T67849 D0C9JZ 58111426 IC50 = 3.4 nM T67849 D0E0YY 53235521 IC50 < 50 nM T67849 D05HIJ 135565159 IC50 = 468 nM T67849 D09SFV 3973 IC50 = 500 nM T67849 D0D0QA 44137675 IC50 = 80 nM T67849 D0P1JI 312145 IC50 = 4 nM T67849 C3FRX9 131989 IC50 = 65700 nM T67849 C05RDN 566479 IC50 = 6800 nM T67849 CY3D4G 617191 IC50 = 3887 nM T67849 CS5O7B 622000 IC50 > 40000 nM T67849 CXC3V1 622262 IC50 = 701 nM T67849 CU73NO 736009 IC50 > 83300 nM T67849 C0L5VC 946390 IC50 = 900 nM T67849 CWOQ49 1627922 IC50 = 90 nM T67849 CKCW93 2612441 IC50 > 100000 nM T67849 C09VKD 2816900 IC50 = 36800 nM T67849 CK79GO 2988969 IC50 > 100000 nM T67849 C1O4KS 4416330 IC50 > 25000 nM T67849 CIN5F7 4904109 IC50 <= 10000 nM T67849 C1YJM9 4912089 IC50 > 83300 nM T67849 CE74CV 5059890 IC50 = 100000 nM T67849 C2OZ0W 6484194 IC50 = 18000 nM T67849 CK2IR4 6852165 IC50 = 180 nM T67849 CE1Y8A 9815659 IC50 = 5100 nM T67849 CJ79RC 9879653 IC50 = 3 nM T67849 CC4F8I 10021687 IC50 = 800 nM T67849 CZM84H 10066542 IC50 = 800 nM T67849 C2W9ED 10269329 IC50 = 230 nM T67849 C7SFI1 10296883 IC50 > 10000 nM T67849 C32NQS 10357196 IC50 = 4204 nM T67849 CAZT53 10475366 IC50 = 29 nM T67849 CL8YE3 11230964 IC50 = 2900 nM T67849 C8Y6IM 11234514 IC50 = 98 nM T67849 CK65NF 11418892 Ki = 2900 nM T67849 CL3Z4O 11419728 IC50 = 16 nM T67849 CYBD21 11428504 IC50 = 140 nM T67849 CI2YV6 11474717 IC50 = 197 nM T67849 CHJ30L 11492951 IC50 > 20000 nM T67849 CR41FO 11502414 IC50 = 6 nM T67849 C0O4SQ 11522078 IC50 > 5000 nM T67849 C7HMO6 11526786 IC50 = 11 nM T67849 C38YWS 11541283 IC50 = 1 nM T67849 C1VA4C 11543481 IC50 = 810 nM T67849 CN2MS6 11562853 IC50 = 25.12 nM T67849 CMVQ43 11576772 IC50 = 0.9 nM T67849 C8K6VJ 11584055 Ki = 1.1 nM T67849 CEHZ82 11599141 IC50 = 39.81 nM T67849 C1ZPM5 11630874 IC50 = 20000 nM T67849 CYU3J9 11634899 IC50 = 1.7 nM T67849 CP04JC 11666231 IC50 = 16.1 nM T67849 C48YXV 11677284 Ki = 4.9 nM T67849 CY8C9P 11751126 IC50 = 201 nM T67849 CBR6D5 11955693 IC50 = 187 nM T67849 C60DBM 11998444 IC50 = 31710 nM T67849 C5FTB0 11998445 IC50 = 1176 nM T67849 C68WMR 11998447 IC50 = 26240 nM T67849 CYL24B 11998448 IC50 = 5973 nM T67849 CNPI54 11998563 IC50 = 2525 nM T67849 C6AK0Y 11998564 IC50 = 1392 nM T67849 CMVA72 11998565 IC50 = 126 nM T67849 CJ3YP8 11998685 IC50 = 2124 nM T67849 CV8PB5 11998690 IC50 = 614 nM T67849 CB9T1H 11998803 IC50 = 35 nM T67849 C59SKD 11999032 IC50 = 18 nM T67849 CY7A0T 14638904 IC50 = 12500 nM T67849 CH1DJ6 16036739 IC50 = 16 nM T67849 CVN8B2 16049456 IC50 = 251.19 nM T67849 CW2XK6 16050925 IC50 = 530 nM T67849 CW5FD8 16081736 IC50 = 1482 nM T67849 CV9US5 16736978 IC50 = 5300 nM T67849 CF6JS9 16757570 IC50 = 340 nM T67849 CB19TH 16757576 IC50 = 1000 nM T67849 C1NZC7 16757579 IC50 = 166 nM T67849 C1SN9M 17756679 IC50 >= 100000 nM T67849 CVDL81 22036885 IC50 = 0.65 nM T67849 C61ZGT 22135435 IC50 = 79432.82 nM T67849 CP05ZB 22346757 IC50 = 23000 nM T67849 C1F2TM 23582995 IC50 = 950 nM T67849 CEYL29 23585510 Ki = 740 nM T67849 COW91A 23586721 IC50 = 710 nM T67849 CBL37C 23642173 Ki = 4 nM T67849 C8J1SI 23642272 IC50 = 722 nM T67849 C29SFI 24768579 IC50 = 249 nM T67849 C72BSE 24804168 IC50 = 19952.62 nM T67849 C6Y5GV 24805152 IC50 = 19952.62 nM T67849 CL4C8H 24809743 IC50 = 3600 nM T67849 CP4G9Z 24855584 Ki = 3 nM T67849 CJV7D9 24855887 IC50 = 54 nM T67849 CM9C0R 24866805 IC50 = 6700 nM T67849 CB79YC 24905143 IC50 = 250 nM T67849 C2DC9J 24905144 IC50 = 800 nM T67849 CN6V8Z 24905145 IC50 = 27 nM T67849 CSB7P5 24905148 IC50 = 2300 nM T67849 CGSF21 24905149 IC50 = 3 nM T67849 CVDG02 24905150 IC50 = 10200 nM T67849 CWH6C5 24905152 IC50 = 6 nM T67849 C0HE2Q 24905153 IC50 = 4 nM T67849 C7QSC9 24905154 IC50 = 680 nM T67849 CO9D0K 24905155 IC50 = 410 nM T67849 C5W9UR 24905157 IC50 = 140 nM T67849 CC1DA3 24905158 IC50 = 690 nM T67849 COW79F 24905159 IC50 = 650 nM T67849 CFPA53 24905160 IC50 = 640 nM T67849 C2O0JX 24905161 IC50 = 1400 nM T67849 CA72BE 24905162 IC50 = 210 nM T67849 CQN6X9 24905163 IC50 = 1900 nM T67849 CD4O1F 24905165 IC50 = 3700 nM T67849 CKL48T 24905166 IC50 = 1200 nM T67849 C76VYL 24905167 IC50 = 900 nM T67849 C7K5PU 24905168 IC50 = 125 nM T67849 CZ57ID 24905169 IC50 = 730 nM T67849 C2DHX9 24905170 IC50 = 1900 nM T67849 CSB96E 24905171 IC50 = 100000 nM T67849 CWZ0R2 24905172 IC50 = 1300 nM T67849 CY3B6M 24905175 IC50 = 281 nM T67849 CW1V0H 24905177 IC50 = 1900 nM T67849 CO6Y0L 24905178 IC50 = 37000 nM T67849 C60NQW 24905179 IC50 = 686 nM T67849 C4MO8B 24905180 IC50 = 677 nM T67849 COJI47 24905181 IC50 = 249 nM T67849 CS0B2C 24905182 IC50 = 72 nM T67849 C1H4BT 24905183 IC50 = 144 nM T67849 C4WHK9 24905184 IC50 = 2970 nM T67849 C7Q4MZ 24905185 IC50 = 2480 nM T67849 CS4IP1 24905186 IC50 = 130 nM T67849 C69QWO 24905187 IC50 = 1030 nM T67849 C85ANB 24905188 IC50 = 173 nM T67849 CNHD75 24905189 IC50 = 57 nM T67849 C9JUO2 24905190 IC50 = 2020 nM T67849 CPR03K 24905191 IC50 = 446 nM T67849 CTAG19 24905193 IC50 = 228 nM T67849 C7VJM5 24905194 IC50 = 643 nM T67849 CEP1L3 24905195 IC50 = 436 nM T67849 CP68ZD 24905196 IC50 = 429 nM T67849 C8Z0RJ 24905197 IC50 = 255 nM T67849 CN9RT0 24905198 IC50 = 1200 nM T67849 CHI78P 24905200 IC50 = 400 nM T67849 CO6PE8 24905201 IC50 = 340 nM T67849 CZ63HS 24905202 IC50 = 77 nM T67849 C2X0FC 24905203 IC50 = 120 nM T67849 C0WCE3 24905204 IC50 = 90 nM T67849 CNK50B 24905205 IC50 = 89 nM T67849 C12DPB 24905206 IC50 = 190 nM T67849 C8N0RH 24905207 IC50 = 3700 nM T67849 CYA5G2 24905208 IC50 = 56 nM T67849 CDV2B4 24905209 IC50 = 660 nM T67849 CEFK68 24905210 IC50 = 140 nM T67849 CUFP12 24905211 IC50 = 453 nM T67849 C0JG8L 24905212 IC50 = 966 nM T67849 CP47MK 24905213 IC50 = 18000 nM T67849 CB61QC 24905214 IC50 = 2300 nM T67849 CQ13ZI 24905215 IC50 = 3400 nM T67849 C6VI8F 24905216 IC50 = 123 nM T67849 CXNH25 24905217 IC50 = 85 nM T67849 C2PN9S 24905218 IC50 = 49 nM T67849 C9O2AL 24905219 IC50 = 110 nM T67849 CIT7U8 24905220 IC50 = 1800 nM T67849 CMD26S 24905221 IC50 = 37 nM T67849 C4R8WC 24905222 IC50 = 443 nM T67849 C47SHA 24905223 IC50 = 100 nM T67849 C1DY2R 24905224 IC50 = 142 nM T67849 CS0XF9 24905225 IC50 = 409 nM T67849 CG5VX2 24905226 IC50 = 100000 nM T67849 C57QEO 24905227 IC50 = 100000 nM T67849 C7CG5E 24905228 IC50 = 1000 nM T67849 CHP5D1 24905229 IC50 = 1700 nM T67849 CXP09S 24905230 IC50 = 120 nM T67849 CY7XG1 24905231 IC50 = 1500 nM T67849 C7JFQ2 24905232 IC50 = 375 nM T67849 C2JM1P 24905233 IC50 = 5200 nM T67849 CC3BF0 24905234 IC50 = 3900 nM T67849 CE57FI 24905235 IC50 = 3900 nM T67849 CUP20O 24905236 IC50 = 6300 nM T67849 CLC6Q2 24905237 IC50 = 1400 nM T67849 C9M1GI 24905238 IC50 = 213 nM T67849 CVD72F 24905239 IC50 = 68 nM T67849 CK38IZ 24905240 IC50 = 88 nM T67849 CO2V5E 24905241 IC50 = 2000 nM T67849 CZBA19 24905244 IC50 = 162 nM T67849 CQ8OI1 24905246 IC50 = 72000 nM T67849 C5URC6 24905247 IC50 = 1800 nM T67849 CZ2E9K 24905249 IC50 = 3000 nM T67849 C03SVO 24905250 IC50 = 9600 nM T67849 CIF2J5 24905251 IC50 = 280 nM T67849 CPTE58 24905252 IC50 = 1260 nM T67849 CX1JB8 24905253 IC50 = 5700 nM T67849 COZ3H7 24905254 IC50 = 29000 nM T67849 CDT1H9 24905255 IC50 = 11000 nM T67849 C54QKA 24905256 IC50 = 3100 nM T67849 CRU3P2 24905257 IC50 = 100000 nM T67849 C9U0JA 24905259 IC50 = 11000 nM T67849 CO4YS7 24905260 IC50 = 82000 nM T67849 CEG0B5 24905261 IC50 = 100000 nM T67849 C9VE5F 24905262 IC50 = 100000 nM T67849 C3I4HK 24905264 IC50 = 6300 nM T67849 C0VMI6 24905265 IC50 = 100000 nM T67849 CWE3V0 24905267 IC50 = 100000 nM T67849 CH4T3A 24905268 IC50 = 100000 nM T67849 CVT17Q 24905270 IC50 = 750 nM T67849 C6QDN7 24905271 IC50 = 2900 nM T67849 C6XHJ7 24905272 IC50 = 1200 nM T67849 CTB9A3 24905273 IC50 = 28000 nM T67849 C0NB1Q 24905274 IC50 = 21000 nM T67849 C9KQ0L 24905275 IC50 = 3000 nM T67849 C9O8QZ 24905277 IC50 = 7400 nM T67849 CP50RD 24905280 IC50 = 65 nM T67849 CG13ZM 24905281 IC50 = 252 nM T67849 CF0S6X 24905282 IC50 = 42 nM T67849 C5HBL0 24905284 IC50 = 3190 nM T67849 C2Z5DN 24905285 IC50 = 660 nM T67849 CL6GH8 24905286 IC50 = 198 nM T67849 CKYO98 24905287 IC50 = 220 nM T67849 CRNQ65 24905288 IC50 = 74 nM T67849 COD7I5 24905289 IC50 = 470 nM T67849 C4LP7E 24905290 IC50 = 210 nM T67849 CE9JC2 24905291 IC50 = 76 nM T67849 C2GI1R 24905292 IC50 = 473 nM T67849 CHW8C4 24905293 IC50 = 47 nM T67849 CQF0H1 24905294 IC50 = 10 nM T67849 CNO7X0 24905295 IC50 = 12 nM T67849 C5WRG7 24905296 IC50 = 17 nM T67849 CQ1S0U 24905297 IC50 = 276 nM T67849 C4UES7 24905298 IC50 = 177 nM T67849 CMS69P 24905299 IC50 = 6050 nM T67849 CC0U5M 24905300 IC50 = 103 nM T67849 CW7X6S 24905301 IC50 = 1985 nM T67849 C97IQV 24905302 IC50 = 142 nM T67849 CSJ47V 24905303 IC50 = 199 nM T67849 CPN74C 24905304 IC50 = 5470 nM T67849 C5CS3N 24905305 IC50 = 207 nM T67849 CK4XE9 24905307 IC50 = 172 nM T67849 CTU6Z3 24905308 IC50 = 1070 nM T67849 C9SQX1 24905309 IC50 = 193 nM T67849 CM75JP 24905310 IC50 = 514 nM T67849 C9Q2BJ 24905311 IC50 = 680 nM T67849 C9VUA1 24905312 IC50 = 203 nM T67849 CU3RS1 24905313 IC50 = 215 nM T67849 CYG3H2 24905314 IC50 = 213 nM T67849 CV5Q7O 24905315 IC50 = 58 nM T67849 C8SA3O 24905316 IC50 = 13 nM T67849 CI5MN3 24905317 IC50 = 20 nM T67849 CJ1P7K 24905318 IC50 = 12 nM T67849 C1T6YQ 24905319 IC50 = 15 nM T67849 CAU86X 24905320 IC50 = 49 nM T67849 C54ISY 24905321 IC50 = 3030 nM T67849 C2GE5I 24905322 IC50 = 1620 nM T67849 C8D6YK 24905323 IC50 = 4350 nM T67849 C5NZH9 24905324 IC50 = 1000 nM T67849 C9D6JR 24905325 IC50 = 777 nM T67849 CLZT41 24905326 IC50 = 150 nM T67849 CW8FD3 24905327 IC50 = 74 nM T67849 CHB7A2 24905328 IC50 = 1370 nM T67849 CA8EI3 24905329 IC50 = 716 nM T67849 CCQ0O7 24905330 IC50 = 197 nM T67849 CJ81AS 24905331 IC50 = 23 nM T67849 C8PW4H 24905332 IC50 = 41 nM T67849 C2Y5TF 24905333 IC50 = 112 nM T67849 CH9FL5 24905334 IC50 = 67 nM T67849 C1S0PC 24905335 IC50 = 120 nM T67849 C8N9MV 24905336 IC50 = 206 nM T67849 C9E8BJ 24905338 IC50 = 240 nM T67849 CX85AC 24905341 IC50 = 6900 nM T67849 CKZ80E 24905342 IC50 = 46 nM T67849 CO8SH1 24905343 IC50 = 48 nM T67849 C7IZL6 24905344 IC50 = 670 nM T67849 C43VSW 24936353 IC50 = 10 nM T67849 C83EUF 24937010 IC50 = 3 nM T67849 C72LWC 24937637 IC50 = 3.2 nM T67849 C6E3AN 24944519 IC50 = 0.5 nM T67849 CHI9W6 24944522 IC50 = 105.9 nM T67849 C98MEW 24946175 IC50 = 11 nM T67849 CC7H3U 24946706 IC50 = 0.7 nM T67849 C78NJE 24955795 IC50 = 549 nM T67849 C8P6NT 24956158 IC50 = 80 nM T67849 CJI29P 24956159 IC50 = 5731 nM T67849 CXV6R0 24968746 Ki = 7 nM T67849 C6C4RH 24993871 IC50 = 12 nM T67849 CEW91Q 25032963 IC50 = 4 nM T67849 CY50OT 25052783 IC50 = 32 nM T67849 CHR51O 25057242 IC50 = 61 nM T67849 CF8G3J 25095512 IC50 = 2 nM T67849 CD69RK 25097993 IC50 < 0.5 nM T67849 CLP07J 25110819 IC50 > 10000 nM T67849 CVM89J 25128663 IC50 = 5011.87 nM T67849 C4HRL9 25128667 IC50 = 1995.26 nM T67849 C4SWT5 25128668 IC50 > 79432.82 nM T67849 CIO6A4 25129024 IC50 > 100000 nM T67849 CLS7P0 25129381 IC50 = 6309.57 nM T67849 C9R2EA 25129383 IC50 = 31622.78 nM T67849 C4YZL9 25129386 IC50 = 5011.87 nM T67849 CDO9Q0 25129729 IC50 > 100000 nM T67849 CX86YV 25129734 IC50 > 19952.62 nM T67849 CA2K4U 25130429 IC50 = 501.19 nM T67849 C1J8KH 25132804 IC50 = 3162.28 nM T67849 CI04XW 25132806 IC50 = 31622.78 nM T67849 C5WC4L 25133141 IC50 > 31622.78 nM T67849 CSH37X 25133142 IC50 > 10000 nM T67849 CW3HN6 25133144 IC50 > 100000 nM T67849 C4LHV1 25165368 IC50 > 10000 nM T67849 C2CXH3 25165371 IC50 > 10000 nM T67849 CQWL59 25165372 IC50 > 10000 nM T67849 CL87JW 25165773 IC50 > 30000 nM T67849 CB89TL 25165774 IC50 > 10000 nM T67849 CFZI92 25165961 IC50 > 10000 nM T67849 CK2YI4 25168990 IC50 = 9332.54 nM T67849 C7G1ZM 25169579 IC50 = 250 nM T67849 CL81FJ 25169580 IC50 = 320 nM T67849 C8WL0Z 25169784 IC50 > 1000 nM T67849 CLR8M2 25169786 IC50 = 690 nM T67849 CL3UK2 25170000 IC50 > 1000 nM T67849 C6WCR7 25170003 IC50 = 120 nM T67849 C2RT9W 25170004 IC50 = 230 nM T67849 CSK97U 25170005 IC50 > 1000 nM T67849 C7AH2I 25170203 IC50 = 280 nM T67849 C2TEW6 25170204 IC50 > 1000 nM T67849 C5PTZ0 25170410 IC50 = 89 nM T67849 CLJR80 25171641 IC50 = 3400 nM T67849 C7ZQC2 25171642 IC50 = 700 nM T67849 C7AHP4 25171644 IC50 > 1000 nM T67849 CX6BL8 25171852 IC50 > 1000 nM T67849 C7TL2N 25171853 IC50 > 1000 nM T67849 C6BR3F 25171855 IC50 = 90 nM T67849 CMI85O 25171856 IC50 = 150 nM T67849 CUN9F3 25171857 IC50 = 170 nM T67849 CKY81J 25172061 IC50 > 1000 nM T67849 CC1D8V 25172062 IC50 = 49 nM T67849 C1L6GX 25172063 IC50 = 410 nM T67849 CFO08N 25172065 IC50 = 35 nM T67849 C8ZF0A 25172066 IC50 = 2000 nM T67849 CCW80B 25172270 IC50 > 1000 nM T67849 C9HUB6 25172271 IC50 = 310 nM T67849 CC60ZY 25172272 IC50 = 180 nM T67849 C54EGX 25172274 IC50 = 400 nM T67849 C5QVC7 25172275 IC50 = 200 nM T67849 CPW2D9 25172477 IC50 = 54 nM T67849 CVDC60 25172479 IC50 = 580 nM T67849 CI6W9H 25172661 IC50 = 9.3 nM T67849 CL5IC0 25172662 IC50 = 110 nM T67849 CDAO95 25172663 IC50 = 180 nM T67849 C8JC3P 25172664 IC50 = 8.6 nM T67849 CK38ER 25172665 IC50 = 16 nM T67849 C3JI1Y 25172666 IC50 = 37 nM T67849 CLW96O 25207689 IC50 = 6 nM T67849 CWP29U 25242324 IC50 = 16 nM T67849 C96OGS 25260915 IC50 = 64 nM T67849 CUR93V 25261554 IC50 > 10000 nM T67849 C3IDN0 25266674 IC50 = 1000 nM T67849 C2IM0O 39733146 IC50 = 7943.28 nM T67849 C1O8ZY 42596976 IC50 = 665 nM T67849 CO4PL8 42606076 IC50 > 100000 nM T67849 C20VGT 42606077 IC50 = 39000 nM T67849 C7N5EC 42606078 IC50 > 100000 nM T67849 CIF63E 42623219 IC50 = 6309.57 nM T67849 C3DNM9 42623223 IC50 = 1584.89 nM T67849 COR5I0 42623224 IC50 = 7943.28 nM T67849 CX1DC2 42623385 IC50 = 398.11 nM T67849 CR6N3I 42623632 IC50 > 6309.57 nM T67849 C4EM0W 42623869 IC50 = 1584.89 nM T67849 C5TY9Q 42623950 IC50 = 3162.28 nM T67849 C10RBA 42636535 IC50 = 1500 nM T67849 CKH08W 44123663 IC50 < 100 nM T67849 C3ROX1 44124863 Ki = 0.8 nM T67849 CI3K7H 44129042 IC50 = 4000 nM T67849 CIE0J3 44129043 IC50 = 7900 nM T67849 CUW85V 44129044 IC50 > 10000 nM T67849 C2B9DE 44129118 IC50 = 3800 nM T67849 C0R1PH 44129198 IC50 = 8100 nM T67849 C6LGD5 44129200 IC50 = 630 nM T67849 C03RLS 44129270 IC50 > 10000 nM T67849 CU4H1I 44129274 IC50 = 7400 nM T67849 C79QOC 44129275 IC50 = 1600 nM T67849 C0W3ZF 44129348 IC50 = 9200 nM T67849 CH6RO4 44129351 IC50 = 3300 nM T67849 CPAU59 44129353 IC50 = 1800 nM T67849 CN5O4I 44129429 IC50 = 810 nM T67849 C3ZSV2 44129432 IC50 = 1500 nM T67849 CM5U2I 44137407 IC50 = 190 nM T67849 CF17OS 44180029 IC50 = 4200 nM T67849 CHK8Z6 44180034 IC50 = 27 nM T67849 CEJ5F7 44180035 IC50 > 20000 nM T67849 CQNT23 44180155 IC50 > 50000 nM T67849 CIKM57 44180156 IC50 = 960 nM T67849 CBP2T3 44180157 IC50 = 7894 nM T67849 C9CGB4 44180282 IC50 > 50000 nM T67849 C2S5LC 44180395 IC50 = 26 nM T67849 C40NOQ 44180397 IC50 = 18 nM T67849 CTB46H 44180398 IC50 = 12 nM T67849 CE30IL 44180626 IC50 = 20 nM T67849 CRS2G3 44180853 IC50 = 14940 nM T67849 C2VZX7 44181492 IC50 = 2420 nM T67849 C7SYM2 44181493 IC50 > 50000 nM T67849 CB8KF1 44181494 IC50 > 23000 nM T67849 C5AI8R 44181598 IC50 > 30000 nM T67849 CK03RW 44181599 IC50 > 50000 nM T67849 CXL61J 44181600 IC50 = 784 nM T67849 C6TZK5 44181601 IC50 = 481 nM T67849 CCIV74 44181602 IC50 = 555 nM T67849 C36WUP 44181603 IC50 > 50000 nM T67849 CS2U7R 44181604 IC50 = 9807 nM T67849 CL6W0C 44181605 IC50 = 8936 nM T67849 CFD41Z 44181718 IC50 = 13830 nM T67849 C2RB1P 44181719 IC50 > 23000 nM T67849 CMC75I 44181720 IC50 = 1142 nM T67849 CWTS93 44181721 IC50 = 3998 nM T67849 CT1JL2 44181722 IC50 = 3732 nM T67849 CE9HO1 44181723 IC50 = 278 nM T67849 CFSB29 44181724 IC50 = 649 nM T67849 C13DKP 44219291 IC50 = 12 nM T67849 CMNC52 44225402 IC50 < 50 nM T67849 C6RDB9 44237450 IC50 > 100 nM T67849 C98MAL 44436951 IC50 = 5400 nM T67849 CD0ME6 44436952 IC50 > 10000 nM T67849 CR6ZU9 44436953 IC50 > 10000 nM T67849 CYK0T1 44436954 IC50 > 10000 nM T67849 CYV15O 44436955 IC50 > 10000 nM T67849 C3M4RN 44436961 IC50 > 10000 nM T67849 CA4SV2 44436964 IC50 > 10000 nM T67849 CO5FK1 44436967 IC50 > 10000 nM T67849 CRKU98 44436970 IC50 > 10000 nM T67849 C9V1SZ 44436971 IC50 > 10000 nM T67849 CZ4V2L 44436972 IC50 > 10000 nM T67849 COG34Q 44436976 IC50 > 10000 nM T67849 C4RAK8 44436979 IC50 = 9000 nM T67849 CXN93Q 44436980 IC50 > 10000 nM T67849 CX57RI 44436981 IC50 > 10000 nM T67849 C9ZML1 44454396 IC50 = 35 nM T67849 C4PR1L 44466962 Ki = 10 nM T67849 C30NZA 44475985 IC50 = 21 nM T67849 CAT8F7 44475986 IC50 = 1 nM T67849 CSR73H 44475987 IC50 = 7 nM T67849 CDAX92 44475988 IC50 = 40 nM T67849 CBH0S5 44475989 IC50 = 34 nM T67849 CW5A7L 44475990 IC50 = 0.5 nM T67849 CG9A5L 44511405 IC50 <= 10000 nM T67849 CFC65B 44539960 IC50 <= 10000 nM T67849 C03IGD 44540030 IC50 = 1584.89 nM T67849 C5LWU1 44540126 IC50 = 3981.07 nM T67849 CYD4Z8 44540130 IC50 = 1.995 nM T67849 CAT2R7 44540316 IC50 = 3162.28 nM T67849 C36NRP 44540403 IC50 <= 10000 nM T67849 C2T9GC 44540407 IC50 = 100 nM T67849 CQ4PE7 44540492 IC50 = 1000 nM T67849 CZ9GL8 44541044 IC50 = 12.59 nM T67849 C6L4SV 44545041 Ki = 4 nM T67849 CPCJ61 44554231 IC50 < 100 nM T67849 C0N2VK 44554233 IC50 < 100 nM T67849 C3VRO9 44557921 IC50 = 707.95 nM T67849 CN2O9S 44577591 IC50 > 20000 nM T67849 CRE61W 44577592 IC50 = 74 nM T67849 CH63GM 44577593 IC50 = 20 nM T67849 CA8MV5 44577594 IC50 = 153 nM T67849 C9IXW8 44577638 IC50 = 94 nM T67849 C8A5RT 44577639 IC50 = 21 nM T67849 CNP02V 44577640 IC50 = 26 nM T67849 CT6GN5 44577641 IC50 = 123 nM T67849 CIQR97 44577850 IC50 = 1631 nM T67849 CCG8P9 44577851 IC50 = 11240 nM T67849 CNF47Q 44577852 IC50 = 15280 nM T67849 CLBA40 44577853 IC50 = 783 nM T67849 COU6V7 44577854 IC50 = 605 nM T67849 C8M5FY 44577914 IC50 = 366 nM T67849 C3MGZ9 44577915 IC50 = 1050 nM T67849 CGO09K 44577916 IC50 = 50 nM T67849 CRJ3B7 44577917 IC50 = 155 nM T67849 CTR89C 44577918 IC50 = 7574 nM T67849 CO05YG 44577919 IC50 = 81 nM T67849 CT70WA 44577920 IC50 = 17 nM T67849 C5KXS4 44577921 IC50 = 90 nM T67849 CZ2HI5 44577922 IC50 = 51 nM T67849 CGTU34 44577950 IC50 = 285 nM T67849 CQC50R 44577951 IC50 = 49 nM T67849 C8ZTW2 44577952 IC50 = 230 nM T67849 CIL93G 44577953 IC50 = 357 nM T67849 C8NB5H 44578037 IC50 > 40000 nM T67849 CX9TO2 44578038 IC50 = 19040 nM T67849 C7AHR4 44578039 IC50 > 50000 nM T67849 C13LGI 44578040 IC50 > 50000 nM T67849 CNZ06H 44578074 IC50 > 50000 nM T67849 C41TYA 44578108 IC50 = 74 nM T67849 C2W3SQ 44578109 IC50 = 60 nM T67849 CYM69I 44580064 IC50 = 9 nM T67849 CV09JM 44580065 IC50 = 21 nM T67849 CF37TO 44580066 IC50 = 30 nM T67849 CA0BU6 44580067 IC50 = 245 nM T67849 COQ85J 44580235 IC50 = 12 nM T67849 CD4ER0 44580236 IC50 = 7 nM T67849 CHVQ28 44580237 IC50 = 6 nM T67849 C8N2AF 44580238 IC50 = 103 nM T67849 C40LVX 44580274 IC50 = 231 nM T67849 CO9LD8 44580275 IC50 = 103 nM T67849 C5QWG4 44580276 IC50 = 89 nM T67849 CFZS45 44580277 IC50 = 72 nM T67849 CQ4CR6 44580635 IC50 = 32 nM T67849 CJHK57 44580636 IC50 = 65 nM T67849 CC6M2E 44580684 IC50 = 17 nM T67849 CA3KP5 44580685 IC50 = 43 nM T67849 C40VHS 44580686 IC50 = 14 nM T67849 CXV92J 44580687 IC50 = 29 nM T67849 CG3PH2 44580721 IC50 = 45 nM T67849 CIO46B 44580722 IC50 = 4 nM T67849 CNLS71 44580723 IC50 = 4 nM T67849 C1N0MF 44580724 IC50 = 8 nM T67849 CAHQ76 44580766 IC50 = 39 nM T67849 C2XN6B 44580767 IC50 = 4 nM T67849 CC36YN 44580768 IC50 = 36 nM T67849 CZ56FY 44580769 IC50 = 14 nM T67849 C0L2HO 44593630 IC50 = 139 nM T67849 C2NQ6Z 44593631 IC50 = 16 nM T67849 CY3SV7 44596118 IC50 > 10000 nM T67849 C47FHE 44608747 IC50 < 30 nM T67849 CH6V9F 44608754 IC50 = 6 nM T67849 C0IY9N 44608757 IC50 = 6 nM T67849 C90ITS 44608915 IC50 = 4.3 nM T67849 CZH1P9 44609387 IC50 = 4.4 nM T67849 CNDX48 44609388 IC50 = 5.6 nM T67849 C2ISK4 44610761 IC50 = 47000 nM T67849 CE95RQ 44620964 IC50 = 1.4 nM T67849 CVYJ36 44620965 IC50 = 6.6 nM T67849 CA8BY7 44621440 IC50 < 19952623.15 nM T67849 C5M1FR 44621441 IC50 = 31622776.6 nM T67849 C5LD7E 44621442 IC50 = 12589254.12 nM T67849 CO4GT0 44621447 IC50 = 25118864.32 nM T67849 CUV26H 44621448 IC50 = 7943282.35 nM T67849 CV2MG9 44621449 IC50 = 31622776.6 nM T67849 C24IYW 44621451 IC50 = 25118864.32 nM T67849 C0F9YW 44621452 IC50 = 19952623.15 nM T67849 C0GRD8 44621454 IC50 = 39810717.06 nM T67849 C4YHJ0 44621456 IC50 = 31622776.6 nM T67849 C31VBF 44621458 IC50 = 7943282.35 nM T67849 CZ68MG 45488079 IC50 = 945 nM T67849 CV1U7I 46180604 IC50 = 2.4 nM T67849 CED2B3 46180606 IC50 = 310 nM T67849 CDV85O 46180663 IC50 = 100 nM T67849 CZGB46 46180666 IC50 = 5.2 nM T67849 CAU17V 46202808 IC50 = 79.43 nM T67849 CDA3R9 46220225 IC50 = 11 nM T67849 CM82RF 46239494 IC50 = 9 nM T67849 C7RF5Y 46239967 IC50 = 440 nM T67849 C9Z4HV 46830931 IC50 = 676 nM T67849 CIU7W9 46831535 IC50 = 11 nM T67849 CH59DF 46832094 IC50 > 1000 nM T67849 CD05UP 46832357 IC50 = 292 nM T67849 C94YRI 46853654 IC50 = 15.85 nM T67849 C45JIE 46861590 Ki = 3 nM T67849 CZ3WS1 46861592 IC50 = 0.4 nM T67849 CQ2Y1V 46866705 Ki = 0.122 nM T67849 C63RCG 46870269 IC50 = 12.59 nM T67849 CTQ25M 46871497 IC50 = 63.1 nM T67849 CV96TI 46871579 IC50 < 100 nM T67849 CQB16A 46872415 IC50 > 20000 nM T67849 C3HMQ2 46891474 IC50 = 0.6 nM T67849 CB6Z8P 46892208 IC50 = 5800 nM T67849 CZX46Y 46892342 IC50 = 890 nM T67849 C5FN6I 46892845 IC50 = 510 nM T67849 CQ32BN 46892970 IC50 = 3 nM T67849 COJA32 46892971 Ki = 11 nM T67849 C5QFB3 46893088 IC50 = 320 nM T67849 CS30AI 46893754 IC50 = 4000 nM T67849 CJ0VB4 46932297 IC50 = 330 nM T67849 CF14PE 46947264 IC50 = 77 nM T67849 CV90JU 49764911 IC50 = 10000 nM T67849 COE37N 49778924 IC50 = 20 nM T67849 C7ZK3D 49783923 Ki = 0.07943 nM T67849 CHX76J 49784892 Ki = 37 nM T67849 CA1H8S 49784893 Ki = 130 nM T67849 CP2QD0 49784894 Ki = 2 nM T67849 CTZG05 49784988 Ki = 25 nM T67849 CE9AC5 49785078 Ki = 360 nM T67849 CG2IO7 49785079 Ki = 350 nM T67849 C8EYN4 49785083 Ki = 18 nM T67849 CZI34V 49785167 Ki = 810 nM T67849 CJK65T 49785253 Ki = 56 nM T67849 CXK8F5 49785436 Ki = 2 nM T67849 CWL5C6 49785518 Ki = 6 nM T67849 C3NV0J 49785827 Ki = 9 nM T67849 C0OZM2 49785828 Ki = 27 nM T67849 C1AR4G 49785829 Ki = 5000 nM T67849 CA67CQ 49787183 Ki = 0.23 nM T67849 CIR6Z0 49820690 IC50 < 100 nM T67849 CG74VX 49820826 IC50 = 5.6 nM T67849 CKV2N6 49820977 IC50 = 10 nM T67849 CIO24J 49831132 Ki = 5 nM T67849 C50PCV 49831209 Ki = 1.05 nM T67849 C54OBC 49832773 IC50 = 29 nM T67849 C2G0HN 49832939 IC50 = 2.4 nM T67849 C65WEP 49833295 IC50 = 180 nM T67849 C76XBM 49834039 IC50 = 0.67 nM T67849 CGO57N 49834218 IC50 = 3.5 nM T67849 C90JBE 49834576 Ki = 2 nM T67849 CO2LQ5 49834577 IC50 = 19 nM T67849 C5UR4A 49843944 IC50 = 2020 nM T67849 CS40YB 49853846 IC50 = 400 nM T67849 C7PER0 49853953 IC50 = 69 nM T67849 CU9A8O 49854022 IC50 = 1770 nM T67849 C51QVH 49854023 IC50 = 278 nM T67849 CM4HQ2 49854024 IC50 = 2215 nM T67849 C1LBX3 49854049 IC50 = 70 nM T67849 CVC2H6 49854052 IC50 = 64 nM T67849 CC2X9N 49854121 IC50 = 4290 nM T67849 CAJ58E 49854156 IC50 = 110 nM T67849 CAU39Y 49854158 IC50 = 110 nM T67849 CPK6X3 49854360 IC50 = 700 nM T67849 CQ1TZ6 49854365 IC50 = 1600 nM T67849 CJ5I9X 49854461 IC50 = 910 nM T67849 CDXQ69 49854462 IC50 = 5600 nM T67849 C0ORZ9 49854466 IC50 = 1000 nM T67849 CEC10T 49854573 IC50 = 21 nM T67849 C39KQW 49854679 IC50 = 220 nM T67849 C8VDR2 49854680 IC50 = 230 nM T67849 CN2V8R 49854681 IC50 = 970 nM T67849 CSN96A 49855001 IC50 = 390 nM T67849 CALY90 49855192 IC50 = 3900 nM T67849 CJPE20 49855193 IC50 = 1500 nM T67849 CY8MP7 49867926 IC50 = 43 nM T67849 CR0IA5 49871864 IC50 = 8.8 nM T67849 C13WJZ 49872243 IC50 = 1.4 nM T67849 C5OY7B 49872246 IC50 = 0.8 nM T67849 C2KD5E 49872344 IC50 = 1.3 nM T67849 CV5BF3 49872645 IC50 = 1.3 nM T67849 CN97FO 49872646 IC50 = 0.2 nM T67849 CD6P5R 49872735 IC50 = 1.3 nM T67849 CL64NB 49872737 IC50 = 51 nM T67849 CRNG04 49872831 IC50 = 0.8 nM T67849 CQC8B4 49872835 IC50 = 0.6 nM T67849 CPS3O1 49872924 IC50 = 0.4 nM T67849 CUBX74 49872925 IC50 = 0.2 nM T67849 CAW69U 49872927 IC50 = 0.7 nM T67849 CV1L4P 49873242 IC50 = 4.3 nM T67849 C5BA2V 49873243 IC50 = 12 nM T67849 CSN45W 49873329 IC50 = 1.2 nM T67849 C9CW7X 50908894 IC50 = 6 nM T67849 CJ4L8Y 50938829 Ki = 449 nM T67849 CJG65L 50939078 IC50 = 9 nM T67849 CI8QM1 50939080 Ki = 3 nM T67849 CT0IP3 50939081 Ki = 10 nM T67849 C8JD5T 50939209 IC50 = 17 nM T67849 C54EUL 50939212 Ki = 80 nM T67849 CS7Z6U 50939338 IC50 = 6 nM T67849 CXT23Y 50939344 IC50 = 64 nM T67849 C6GH4K 50939865 IC50 = 85 nM T67849 C2I9PS 50939992 IC50 = 362 nM T67849 C9TUE4 50940108 IC50 = 198 nM T67849 CQ93GK 50940110 IC50 = 47 nM T67849 CG4R5C 50940334 IC50 = 626 nM T67849 C2Q0GE 50990922 Ki = 52 nM T67849 CKY3V1 50990924 Ki = 1.2 nM T67849 C5ZF9W 51003380 IC50 = 5100 nM T67849 CY36EH 51003592 IC50 = 794.33 nM T67849 CPA8N1 51039139 Ki > 10000 nM T67849 C6E9WP 51355057 Ki > 10000 nM T67849 C4QE1V 51355058 IC50 = 4000 nM T67849 CO7M9F 51355343 IC50 > 10000 nM T67849 CJ0KM6 51355344 IC50 = 7300 nM T67849 CT0V8F 51355345 Ki > 10000 nM T67849 C0R8XN 51355348 Ki > 10000 nM T67849 C7KT4Z 51355620 Ki > 10000 nM T67849 CI71WE 51355621 Ki = 5147 nM T67849 CLH35Z 51355622 Ki = 7300 nM T67849 CG7T4H 52913198 IC50 = 12 nM T67849 CYU8K9 52913308 IC50 = 4 nM T67849 CD84MT 52913592 IC50 = 110 nM T67849 C2TLG6 52913931 IC50 = 64 nM T67849 CU1P2L 52940797 IC50 = 2400 nM T67849 C2KI6V 52942202 IC50 = 100000 nM T67849 CDHJ08 52942235 IC50 = 490 nM T67849 C4VCY0 52943258 IC50 = 12000 nM T67849 C1XEV2 52943394 IC50 = 156 nM T67849 CHI0P6 52944356 IC50 = 100000 nM T67849 CU16RS 52944387 IC50 = 3600 nM T67849 CWPC54 52945348 IC50 = 125 nM T67849 C4NLX7 52945630 IC50 = 103 nM T67849 CXD6T8 52945845 IC50 = 800 nM T67849 C7ET6Z 52948010 IC50 = 1200 nM T67849 CV5B2C 52949497 IC50 = 15000 nM T67849 C6LFP7 53209481 IC50 = 5.9 nM T67849 CUJ0D4 53209522 IC50 = 2100 nM T67849 C7B4GC 53232894 IC50 <= 10000 nM T67849 CH1Q5D 53234281 IC50 = 3.5 nM T67849 C45JKN 53234283 IC50 = 3.4 nM T67849 C7I6YV 53234922 IC50 < 250 nM T67849 CVK28S 53235062 IC50 < 0.5 nM T67849 COW61E 53235216 IC50 = 2.6 nM T67849 CWE56X 53235217 IC50 = 1.4 nM T67849 CDXM59 53235451 IC50 = 10.2 nM T67849 CD4ZW8 53240744 IC50 <= 10000 nM T67849 CT8IN1 53242225 IC50 = 890 nM T67849 C73RPF 53250077 IC50 = 430 nM T67849 C2UY0C 53252131 IC50 = 13 nM T67849 C4J9WZ 53307606 IC50 = 1.7 nM T67849 C84YNK 53317325 IC50 = 12000 nM T67849 C58NQJ 53318614 IC50 = 43000 nM T67849 C10YUH 53318615 IC50 = 8900 nM T67849 C24GBF 53319075 IC50 = 49 nM T67849 CFJD70 53319932 IC50 = 40800 nM T67849 C3EJB1 53319933 IC50 = 6500 nM T67849 CJRM64 53322563 IC50 = 11100 nM T67849 CN92LK 53322732 IC50 = 20 nM T67849 C23HAU 53361718 IC50 = 5.9 nM T67849 CM60WQ 53361719 IC50 = 6 nM T67849 CL69DK 53377727 IC50 = 29 nM T67849 C6Q8RC 53378051 IC50 = 3.8 nM T67849 CT43IL 53378053 IC50 = 2.6 nM T67849 CBC63U 53378054 IC50 = 27 nM T67849 CF9D0E 53378155 IC50 = 55 nM T67849 C6OQ4K 53378156 IC50 = 6.3 nM T67849 CPWV36 53378900 IC50 = 12 nM T67849 CP4W1Q 53380858 IC50 = 5011.87 nM T67849 CP0ZU1 53465270 IC50 < 100 nM T67849 CNAY79 53482462 Ki = 0.2 nM T67849 CSV9X2 54579940 IC50 = 11 nM T67849 CN51TL 54579941 IC50 = 4600 nM T67849 C7VZU2 54579942 IC50 = 1300 nM T67849 C4R9JB 54579943 IC50 = 690 nM T67849 CG26HQ 54579944 IC50 = 4600 nM T67849 CC5R3O 54580924 IC50 = 240 nM T67849 C3OIY4 54580925 IC50 = 110 nM T67849 C60TYL 54581049 IC50 = 360 nM T67849 CF2UH5 54581983 IC50 = 71 nM T67849 C23EVN 54582916 IC50 = 140 nM T67849 CT2SV7 54583916 IC50 = 40 nM T67849 CY87EC 54583917 IC50 = 710 nM T67849 C8CPI4 54584859 IC50 = 530 nM T67849 C9TZ2V 54584860 IC50 = 3300 nM T67849 CME81Q 54585830 IC50 = 270 nM T67849 CE4TS9 56589559 IC50 = 1.7 nM T67849 CR24WQ 56595421 IC50 = 34 nM T67849 CJ41GT 56595686 IC50 = 2 nM T67849 C2PN4S 56599298 IC50 = 15 nM T67849 CT64SR 56599306 IC50 = 23 nM T67849 CX37YI 56644424 Ki = 0.46 nM T67849 C3S9XF 56645254 Ki = 0.576 nM T67849 CFUT05 56648675 IC50 = 4.3 nM T67849 C1GAB6 56648677 IC50 = 2.4 nM T67849 CWDF40 56648757 IC50 = 1.5 nM T67849 CE35CB 56648758 IC50 = 5.6 nM T67849 CJO39U 56648759 IC50 = 5 nM T67849 C9DX3J 56649281 IC50 = 144 nM T67849 CNKC90 56654649 IC50 = 28 nM T67849 C94JIT 56832510 Ki = 0.61 nM T67849 C0IJP8 56927258 IC50 = 39.81 nM T67849 CM28GU 56928390 IC50 = 12 nM T67849 C9MJG4 56929824 IC50 = 8 nM T67849 CYFB96 56932203 IC50 = 50.12 nM T67849 CJ9R2C 56932209 IC50 = 6309.57 nM T67849 C8C2FG 56932238 IC50 > 19952.62 nM T67849 CX6Q2K 56932240 IC50 = 79.43 nM T67849 C1G4UV 56933328 IC50 < 50 nM T67849 CO6K5Q 56955953 IC50 = 1134 nM T67849 CAK91L 56955954 IC50 = 18 nM T67849 C8B6JG 56955955 IC50 = 816 nM T67849 CW8B4D 57330208 IC50 = 2.4 nM T67849 C6JMN9 57345685 IC50 = 16 nM T67849 CZ7RE0 57345686 IC50 = 7.9 nM T67849 CA53SC 57351276 Ki = 247 nM T67849 CGU27R 57380079 IC50 < 50 nM T67849 C1X3UP 57390135 IC50 > 1000 nM T67849 CQ6N8D 57390136 IC50 = 220 nM T67849 C6XDC8 57390137 IC50 > 1000 nM T67849 C0S6IG 57390138 IC50 = 10 nM T67849 C2RI4V 57390139 IC50 > 1000 nM T67849 CZ3FU2 57390175 IC50 > 1000 nM T67849 CR2X7O 57390176 IC50 > 1000 nM T67849 C1GVK3 57391362 IC50 = 630 nM T67849 C0PR9J 57391364 IC50 = 63 nM T67849 C6L9HO 57391365 IC50 = 20 nM T67849 C2QX0T 57391366 IC50 = 250 nM T67849 CLQ9J1 57391367 IC50 = 13 nM T67849 C53HZJ 57391915 IC50 > 1000 nM T67849 CO18UJ 57391916 IC50 = 900 nM T67849 CRU8Q0 57391917 IC50 = 510 nM T67849 C13DRO 57391952 IC50 > 1000 nM T67849 CH8UV4 57391962 IC50 = 13 nM T67849 CQ1W0C 57393124 IC50 = 50 nM T67849 CZ0RW2 57393125 IC50 = 630 nM T67849 C3G9VK 57393643 IC50 > 1000 nM T67849 CJX56V 57393644 IC50 = 41 nM T67849 CAND02 57393679 IC50 > 1000 nM T67849 CA93ZE 57394864 IC50 = 160 nM T67849 CF6C2T 57395364 IC50 > 1000 nM T67849 CKE35B 57395365 IC50 = 310 nM T67849 CWL2D6 57395366 IC50 > 1000 nM T67849 CB6L7N 57395397 IC50 > 1000 nM T67849 CJH9S2 57395408 IC50 > 1000 nM T67849 C31MCE 57395409 IC50 = 39 nM T67849 CSP45C 57395410 IC50 = 24 nM T67849 CDG2F3 57396625 IC50 = 40 nM T67849 CD73TE 57396626 IC50 = 800 nM T67849 CQRU75 57396627 IC50 = 130 nM T67849 CI34XH 57396628 IC50 = 40 nM T67849 C92FYK 57397192 IC50 = 32 nM T67849 CBC7N6 57397236 IC50 > 1000 nM T67849 CK01SI 57397253 IC50 = 24 nM T67849 C3Q2ZP 57398390 IC50 = 1300 nM T67849 C56TEZ 57398391 IC50 = 200 nM T67849 CP9Q4U 57398392 IC50 = 250 nM T67849 C0O5KE 57398393 IC50 = 16 nM T67849 C5PI3B 57398894 IC50 > 1000 nM T67849 COTK97 57398895 IC50 > 1000 nM T67849 C3G9HW 57399126 IC50 = 630 nM T67849 CYE09F 57400062 IC50 = 20 nM T67849 CN5PY7 57400063 IC50 = 400 nM T67849 CT0Y7E 57400064 IC50 = 160 nM T67849 C0PZM5 57400579 IC50 > 1000 nM T67849 C9BW8C 57400580 IC50 = 100 nM T67849 C4K2RZ 57400581 IC50 > 1000 nM T67849 C4MW8J 57400582 IC50 > 1000 nM T67849 CGC91E 57400641 IC50 = 22 nM T67849 CM63CS 57401865 IC50 = 16 nM T67849 CG6M4H 57401867 IC50 = 400 nM T67849 CP8FY5 57401868 IC50 = 16 nM T67849 CQ5P4X 57401869 IC50 = 80 nM T67849 C2X8PO 57402386 IC50 = 2500 nM T67849 CNMV98 57402387 IC50 = 59 nM T67849 C06IYP 57402428 IC50 = 230 nM T67849 CF68RN 57403576 IC50 = 1000 nM T67849 CL2R7T 57403577 IC50 = 200 nM T67849 CC5N9R 57403578 IC50 = 100 nM T67849 CZ8M5F 57403579 IC50 = 80 nM T67849 C5NT7R 57403580 IC50 = 31 nM T67849 CHBV63 57403581 IC50 = 3 nM T67849 CAC72X 57403582 IC50 = 1300 nM T67849 CNR95F 57404840 IC50 = 2900 nM T67849 CED47A 57410062 IC50 = 133 nM T67849 C1BVX6 57411134 IC50 = 230 nM T67849 C39JSW 57411135 IC50 = 227 nM T67849 CL8F6Q 57411137 IC50 = 435 nM T67849 CW97FT 57411139 IC50 = 485 nM T67849 CU0R3A 57411250 IC50 = 1555 nM T67849 C6C5TU 57411252 IC50 = 2723 nM T67849 CD0W2I 57411254 IC50 = 178 nM T67849 CW1DA3 57411255 IC50 = 1863 nM T67849 C6U4LO 57411256 IC50 = 134 nM T67849 CP9G7L 57411366 IC50 = 567 nM T67849 CC5DO3 57411369 IC50 = 245 nM T67849 C56RBS 57411372 IC50 = 277 nM T67849 CX9O3T 57411485 IC50 = 1000 nM T67849 CQBM65 57411486 IC50 = 483 nM T67849 CK5QX7 57411488 IC50 = 64 nM T67849 C90LNK 57411715 IC50 = 219 nM T67849 CPXE40 57411716 IC50 = 149 nM T67849 CE6RY5 57411836 IC50 = 127 nM T67849 C5JOX3 57411837 IC50 = 58 nM T67849 C0I5JM 57419280 IC50 > 1000 nM T67849 CNI79K 57427669 IC50 = 7943.28 nM T67849 CT6XL0 57466811 Ki = 470 nM T67849 CWOQ10 57494011 IC50 = 3.1 nM T67849 CRB5P2 57495287 IC50 = 23 nM T67849 C59YAC 57495353 IC50 = 79 nM T67849 CMT9L7 57495355 IC50 = 20 nM T67849 CFIY31 57506723 IC50 = 1.8 nM T67849 CUG89V 57506726 IC50 = 0.48 nM T67849 CVOP28 57506727 IC50 = 6 nM T67849 C48BYL 57506732 IC50 = 2.3 nM T67849 CBZS07 57506734 IC50 = 1.8 nM T67849 CK58VZ 57506735 IC50 = 41 nM T67849 CF1KV7 57506736 IC50 = 12 nM T67849 CBQ5X7 57506737 IC50 = 9.8 nM T67849 C1N8DF 57506739 IC50 = 16 nM T67849 CFH0J4 57506741 IC50 = 2.7 nM T67849 CI30AW 57506743 IC50 = 4.3 nM T67849 CL47BS 57506744 IC50 = 2.3 nM T67849 CJE19S 57523686 IC50 = 5715 nM T67849 CUZ31O 57699545 IC50 < 2000 nM T67849 CV9J7D 57748162 IC50 = 1600 nM T67849 CL57CP 57789333 IC50 = 1090 nM T67849 C81BYH 57798309 IC50 = 310 nM T67849 CZ21KP 57900314 IC50 = 3.9 nM T67849 CC60HE 58008590 IC50 = 0.3 nM T67849 CWE7L8 58119648 IC50 = 665 nM T67849 C4MA7Q 58158259 IC50 < 100 nM T67849 CO20YT 58203712 IC50 = 0.6 nM T67849 C7X0OJ 58203779 IC50 = 1.3 nM T67849 CW1M9X 58203976 IC50 = 3.3 nM T67849 COFN62 58203995 IC50 = 8.4 nM T67849 C16GRS 58204034 IC50 = 8.1 nM T67849 CM62NB 58204076 IC50 < 0.5 nM T67849 CGA01N 58204242 IC50 = 1.1 nM T67849 CVR9Q2 58233988 IC50 = 7.943 nM T67849 CB9AH8 58234990 IC50 = 150 nM T67849 CJ8YI2 58234995 IC50 = 90 nM T67849 CZF3U5 58235016 IC50 = 59 nM T67849 CM0ND7 58235018 IC50 = 59 nM T67849 C25RXY 58235020 IC50 = 61 nM T67849 CAY94U 58235030 IC50 = 76 nM T67849 CAJC03 58235033 IC50 = 44 nM T67849 CN7MZ8 58235039 IC50 = 160 nM T67849 CPW84H 58235041 IC50 = 52 nM T67849 C70CRN 58235043 IC50 = 120 nM T67849 C5SQV3 58235052 IC50 = 73 nM T67849 CEZ4T5 58235053 IC50 = 115 nM T67849 C82LIS 58235061 IC50 = 54 nM T67849 C3SO4E 58235062 IC50 = 62 nM T67849 CZ0SD5 58235073 IC50 = 71 nM T67849 CQP25T 58235077 IC50 = 50 nM T67849 C0LDZ2 58235079 IC50 = 110 nM T67849 C2YG5L 58235088 IC50 = 73 nM T67849 C9N7DV 58329366 IC50 < 100 nM T67849 CWYE70 58346211 IC50 = 27 nM T67849 CVHE56 58532021 IC50 = 5 nM T67849 CZEV29 59146228 IC50 < 100 nM T67849 CJ6R8Q 59251679 IC50 = 100 nM T67849 CRZ5B1 59251991 IC50 = 540 nM T67849 CILJ94 59293648 IC50 = 360 nM T67849 C6A3KL 59293676 IC50 = 3000 nM T67849 CC14ZL 59293709 IC50 = 2000 nM T67849 C0R3TX 59293715 IC50 = 960 nM T67849 C9TVC6 59293721 IC50 = 430 nM T67849 CZ5OV1 59293740 IC50 = 2500 nM T67849 CB2Z4R 59293755 IC50 = 1100 nM T67849 C8AL6C 59293763 IC50 = 690 nM T67849 CUVO13 59362157 Ki = 100 nM T67849 CT3CF1 59477024 IC50 > 5011.87 nM T67849 CF6YB8 59477038 IC50 > 100000 nM T67849 CK3H9O 59477041 IC50 = 1258.93 nM T67849 C7KG5E 59477042 IC50 > 39810.72 nM T67849 C01DZW 59477048 IC50 = 1000 nM T67849 C2X8TY 59548177 Ki = 19 nM T67849 CGRO45 59548196 Ki = 60 nM T67849 CD39AG 59548207 Ki > 10000 nM T67849 C6KP4G 59548220 Ki = 63 nM T67849 CTNU85 59548226 Ki = 110 nM T67849 CLB6N4 59548232 Ki = 5700 nM T67849 CSWV07 59548243 Ki = 34 nM T67849 CMT2R0 59548250 Ki = 240 nM T67849 C3I8NE 59548256 Ki = 51 nM T67849 C8W5HT 59548263 Ki = 310 nM T67849 CT8Q5B 59548274 Ki = 7 nM T67849 CVF1B2 59548283 Ki = 62 nM T67849 CY31EA 59548284 Ki = 30 nM T67849 CO4GT7 59548288 Ki = 0.4 nM T67849 CFR7S8 59548302 Ki = 20 nM T67849 CRM20Z 59548320 Ki = 50 nM T67849 CJE5I4 59548341 Ki = 92 nM T67849 C8O1VS 59548349 Ki = 3 nM T67849 CWC65A 59548356 Ki = 3 nM T67849 CMKP95 59548371 Ki = 7 nM T67849 CC8UV3 59548383 Ki = 70 nM T67849 CD4ET2 59548402 Ki = 130 nM T67849 CES59T 59548403 Ki = 300 nM T67849 CE8P3G 59548407 Ki = 6.1 nM T67849 CO4K2W 59548419 Ki = 1.1 nM T67849 CSDB78 59548424 Ki = 4 nM T67849 C81FCQ 59548431 Ki = 6 nM T67849 CLGY34 59548453 Ki = 15 nM T67849 CBT21W 59548454 Ki = 370 nM T67849 CJT68K 59548460 Ki = 39 nM T67849 C9LFT3 59548462 Ki = 1 nM T67849 CX8C2U 59548480 Ki > 10000 nM T67849 C3TU1N 59605243 IC50 = 4 nM T67849 CW4KI5 59605264 Ki = 2 nM T67849 C7F2UV 59605328 IC50 = 2.74 nM T67849 C1OH9X 59605427 IC50 = 23 nM T67849 CAB24G 59605488 IC50 = 3 nM T67849 C09EWP 59605535 Ki = 0.36 nM T67849 CFCQ97 59605669 IC50 = 39 nM T67849 C7U0JF 59605672 IC50 = 7 nM T67849 C5VP8F 59605730 Ki = 0.8 nM T67849 C5B7OK 59605803 IC50 = 1 nM T67849 C8S0ED 59605870 IC50 = 6 nM T67849 C8R0JT 59606002 IC50 = 5.3 nM T67849 CHO01A 59606100 Ki = 1.8 nM T67849 CW9VH5 59606123 Ki = 12.7 nM T67849 C1N8IZ 59606138 IC50 = 2 nM T67849 CYX9T8 59606142 IC50 = 50 nM T67849 C9MEB6 59606148 Ki = 3.1 nM T67849 C4Y3GL 59609976 IC50 = 125 nM T67849 C1PC0J 59634638 IC50 = 2.8 nM T67849 CP2UY3 59634686 IC50 = 2.9 nM T67849 C1TH2N 59634692 IC50 = 8.3 nM T67849 CPA0L2 59634709 IC50 = 3.6 nM T67849 CBI0M6 59688563 IC50 = 25.12 nM T67849 COFZ83 59753763 IC50 = 270 nM T67849 CUYB59 60148924 IC50 = 800 nM T67849 CM8PD7 60150509 IC50 = 4 nM T67849 C5KD3Z 60154714 Ki > 10000 nM T67849 CS0L4D 60154996 Ki > 10000 nM T67849 C1UI3P 60155086 Ki = 6000 nM T67849 CX08ON 60155087 Ki = 910 nM T67849 CX8J1I 60155265 Ki = 10 nM T67849 CAT40I 60155266 Ki = 4 nM T67849 CD56VA 60155268 Ki = 16 nM T67849 CCQB56 60155375 IC50 = 387 nM T67849 CH5X2S 60155376 IC50 = 456 nM T67849 C74FEN 60155377 IC50 = 1095 nM T67849 CZ6G4B 60155378 IC50 = 352 nM T67849 C10AHQ 60155379 IC50 = 1073 nM T67849 C5FI4P 60155451 Ki = 6 nM T67849 CX9G4U 60155452 Ki = 3 nM T67849 C9Q7DE 60155469 IC50 = 638 nM T67849 CH8UY5 60155470 IC50 = 1418 nM T67849 C3EDY4 60155471 IC50 = 1202 nM T67849 CE0ZX1 60155472 IC50 = 1582 nM T67849 CG90MC 60155473 IC50 = 533 nM T67849 C82PVI 60155474 IC50 = 3389 nM T67849 CX49FT 60155475 IC50 = 2964 nM T67849 CR7EG9 60155538 Ki = 21 nM T67849 CU6YB9 60155539 Ki = 13 nM T67849 CW6N1S 60155552 IC50 = 100 nM T67849 CIB08V 60155553 IC50 = 568 nM T67849 CZE28G 60155554 IC50 = 415 nM T67849 CZD2W7 60155555 IC50 = 546 nM T67849 CO6IU3 60155556 IC50 = 1355 nM T67849 C6HN5O 60155557 IC50 = 437 nM T67849 CMQ9G1 60155638 IC50 = 1020 nM T67849 CG56KT 60155639 IC50 = 539 nM T67849 CBJ65P 60155640 IC50 = 1253 nM T67849 C8OJK0 60155641 IC50 = 340 nM T67849 CT9XJ6 60155642 IC50 = 1186 nM T67849 C5BYQ3 60155643 IC50 = 1032 nM T67849 C57RBF 60155722 IC50 = 743 nM T67849 CU7J6L 60155723 IC50 = 2452 nM T67849 CSZA16 60155724 IC50 = 34 nM T67849 C21DWT 60155725 IC50 = 4389 nM T67849 C12CQU 60155726 IC50 = 1316 nM T67849 CA5TM3 60155805 IC50 = 181 nM T67849 C60RIO 60155806 IC50 = 41 nM T67849 CWC26U 60165513 IC50 = 1.1 nM T67849 C67TFB 60165514 IC50 = 134 nM T67849 CPL1G3 60165805 IC50 = 4.3 nM T67849 C54NOW 66552297 IC50 > 100000 nM T67849 CX4HW1 66552298 IC50 > 100000 nM T67849 CEJ54A 66552343 IC50 = 6309.57 nM T67849 CUQ5Y2 66552345 IC50 > 100000 nM T67849 C5F8ZE 66552346 IC50 > 10000 nM T67849 CHQC56 66552347 IC50 > 100000 nM T67849 CS6BQ0 66552348 IC50 > 100000 nM T67849 CGT2V9 66552407 IC50 > 100000 nM T67849 CIJ3C5 66552408 IC50 = 3162.28 nM T67849 C6ZFI1 66552410 IC50 > 100000 nM T67849 C8S7CM 66552411 IC50 > 25118.86 nM T67849 C9A7IK 66552412 IC50 > 100000 nM T67849 CRC24S 66552467 IC50 > 100000 nM T67849 CHU5V3 66552468 IC50 > 100000 nM T67849 C46POH 66552523 IC50 > 100000 nM T67849 C68LXT 66552524 IC50 > 100000 nM T67849 C91JZL 66553214 IC50 = 2210 nM T67849 CUC7B3 66557964 IC50 = 8.6 nM T67849 C9X2TB 66558056 IC50 = 5.1 nM T67849 C5BP3T 66558242 Ki = 2.5 nM T67849 CLR82P 66558244 Ki = 1.7 nM T67849 CUTG05 66558414 Ki = 1.2 nM T67849 C7FKP2 66575655 IC50 = 11 nM T67849 C1R3SI 66653673 IC50 = 358 nM T67849 CF8BZ7 66677439 IC50 = 4 nM T67849 CQ6U8R 66776828 IC50 <= 10000 nM T67849 CN0RE8 66779813 IC50 = 10 nM T67849 C3IP5D 66779815 IC50 = 16 nM T67849 CH86MR 66779905 IC50 = 63 nM T67849 CX2N6E 66779920 IC50 = 320 nM T67849 C9O4TC 66779989 IC50 = 10 nM T67849 CF2UM8 66780001 IC50 = 500 nM T67849 CHU0C5 66780007 IC50 = 3 nM T67849 CGL4V1 66780016 IC50 = 63 nM T67849 C5F6OA 66780027 IC50 = 2000 nM T67849 C8DN7A 66780034 IC50 = 2500 nM T67849 C4AM6R 66780100 IC50 = 13 nM T67849 CZ5P2N 66780118 IC50 = 2 nM T67849 CREA54 66780266 IC50 = 79 nM T67849 CRCA72 66780292 IC50 = 10 nM T67849 CW2SM6 66780337 IC50 = 2 nM T67849 CU54DY 66780379 IC50 = 40 nM T67849 CQ70YA 66780434 IC50 = 160 nM T67849 C8F9UY 66780515 IC50 = 3 nM T67849 CFH6C2 66780644 IC50 = 250 nM T67849 CTZB46 66780835 IC50 > 790 nM T67849 CEP5A2 66780844 IC50 = 500 nM T67849 C51ARE 66788835 Ki = 0.6 nM T67849 C6C8RD 66802145 IC50 = 790 nM T67849 CW12XO 66882257 IC50 = 2400 nM T67849 C6IO1S 66883557 IC50 = 1470 nM T67849 C1HSE0 67035086 IC50 = 120 nM T67849 C38RGB 67035556 IC50 = 6600 nM T67849 C8HOZ9 67041250 IC50 = 4000 nM T67849 C5E4AJ 67050504 IC50 = 7.6 nM T67849 CMWO25 67061712 IC50 < 0.5 nM T67849 C1K5PQ 67094257 Ki = 630 nM T67849 CJ46YU 67094333 Ki = 890 nM T67849 C0OX5N 67103709 IC50 = 41 nM T67849 C9J2EO 67103712 IC50 = 28 nM T67849 CM4W1Y 67103722 IC50 = 32 nM T67849 C5TYQ3 67103909 IC50 = 12 nM T67849 CVJ49E 67103974 IC50 = 53 nM T67849 C3VFY7 67104025 IC50 = 73 nM T67849 CC07KA 67104052 IC50 = 79 nM T67849 C4Z0HT 67159178 IC50 <= 10000 nM T67849 C7EZW6 67192973 IC50 = 82 nM T67849 C1OXI2 67284515 IC50 = 64 nM T67849 CQHF85 67284779 IC50 = 30 nM T67849 C3K4DG 67285093 IC50 = 72 nM T67849 CYD3P9 67285103 IC50 = 450 nM T67849 CT6BX3 67285457 Ki = 154 nM T67849 CY0C7J 67492428 IC50 = 2 nM T67849 C28DWV 67492561 IC50 = 3 nM T67849 CN2Q1E 67492705 IC50 = 5 nM T67849 CEG3F8 67983123 IC50 = 1200 nM T67849 CA18UP 67983576 IC50 > 9100 nM T67849 C8Z0SM 67983581 IC50 = 500 nM T67849 C2Z4HF 67983896 IC50 = 8500 nM T67849 C26TPD 67983918 IC50 = 820 nM T67849 C25AHY 67984037 IC50 = 7000 nM T67849 C7N4ZS 68034365 IC50 = 820 nM T67849 CC19KE 68041083 IC50 = 3.6 nM T67849 C07EHN 68070485 IC50 < 50 nM T67849 C8I7GC 68293638 IC50 > 10000 nM T67849 C19GYQ 68312763 Ki = 0.78 nM T67849 CUN2V4 68312817 Ki = 2.4 nM T67849 CE43WU 68312934 Ki = 2.8 nM T67849 CM19NS 68312957 Ki = 0.88 nM T67849 CAV08T 68313105 Ki = 0.48 nM T67849 C2K0BV 68313143 Ki = 0.81 nM T67849 CR57TQ 68313151 Ki = 1.9 nM T67849 C7TBV6 68498844 IC50 = 94 nM T67849 COQ61U 68501846 IC50 = 680 nM T67849 C4QT2C 68502605 IC50 = 160 nM T67849 CA4LT5 68502607 IC50 = 950 nM T67849 CO5GZ4 68502623 IC50 = 74 nM T67849 CMS39R 68502742 IC50 = 380 nM T67849 C6OUA7 68502808 IC50 = 450 nM T67849 C09HWK 68502836 IC50 = 27 nM T67849 CI1HJ5 68504925 IC50 > 1000 nM T67849 CAB0C1 68505903 IC50 = 350 nM T67849 C01QHM 68547896 IC50 = 200 nM T67849 C53LRM 70673659 IC50 = 210 nM T67849 C0WIT6 70674249 IC50 = 380 nM T67849 C86YWH 70674360 IC50 = 11 nM T67849 C9CZ5S 70674587 IC50 = 18 nM T67849 C45DBH 70674589 IC50 = 7 nM T67849 C0T7CZ 70674590 IC50 = 6.5 nM T67849 C8MTV6 70674592 IC50 = 4.7 nM T67849 C3F7RY 70675053 IC50 = 3 nM T67849 C3BP8R 70675057 IC50 = 6.6 nM T67849 C4XV9C 70675169 IC50 = 76 nM T67849 CAR46Z 70675172 IC50 = 4.6 nM T67849 C16VLO 70675294 IC50 = 51 nM T67849 C97HZQ 70675296 IC50 = 150 nM T67849 CUV7X5 70675427 IC50 = 35 nM T67849 CN09DI 70675846 IC50 = 168 nM T67849 C6BQE1 70681248 IC50 = 40 nM T67849 CPE36T 70681262 IC50 = 25 nM T67849 CPX41V 70682086 IC50 = 25.12 nM T67849 CQW54O 70682591 Ki = 190 nM T67849 CPV59G 70682592 Ki = 1670 nM T67849 CB3ZN5 70683337 IC50 = 130 nM T67849 C1I5PH 70683338 IC50 = 40 nM T67849 CSM0A6 70684204 IC50 = 6.31 nM T67849 CXD08N 70684690 Ki = 74 nM T67849 C8O2QH 70685440 IC50 = 50 nM T67849 CZG9M1 70685441 IC50 = 79 nM T67849 CH7KO0 70685442 IC50 = 25 nM T67849 C6G4WB 70686339 IC50 > 25118.86 nM T67849 CON8X4 70686340 IC50 = 1584.89 nM T67849 C1ASW4 70686341 IC50 = 12.59 nM T67849 C0PWL5 70686455 IC50 = 1258.93 nM T67849 CN4CR2 70686584 IC50 = 260 nM T67849 C85FWA 70686829 Ki = 19 nM T67849 CQS8G7 70686830 Ki = 220 nM T67849 C8QSD2 70688455 IC50 = 15.85 nM T67849 CFCJ02 70688558 IC50 = 19.95 nM T67849 CSX6I7 70688908 Ki = 210 nM T67849 C5YN6U 70689166 IC50 = 500 nM T67849 C6L4WY 70689639 IC50 = 20 nM T67849 CGT1X2 70690496 IC50 = 199.53 nM T67849 CW3U5J 70690994 Ki = 260 nM T67849 CC6I1Q 70691259 IC50 = 1000 nM T67849 CD3JL4 70691776 IC50 = 31 nM T67849 CDK52M 70692650 IC50 = 794.33 nM T67849 CGQJ68 70692914 IC50 > 1000 nM T67849 C7G5UV 70692915 IC50 = 125.89 nM T67849 C3TM1F 70693128 Ki = 79 nM T67849 C2VAU8 70693129 Ki = 61 nM T67849 C65FHO 70694723 Ki = 8 nM T67849 CPFO83 70694805 IC50 = 794.33 nM T67849 CRNY76 70695188 Ki = 79 nM T67849 C3N5YJ 70695189 Ki = 3620 nM T67849 C75YGN 70695469 IC50 = 50 nM T67849 C61CFG 70696737 IC50 = 25.12 nM T67849 C7KL5X 70696852 IC50 = 3162.28 nM T67849 CRH8E2 71270723 IC50 = 25.12 nM T67849 CWR58A 71270783 IC50 = 158.49 nM T67849 CF9LU4 71270807 IC50 = 19.95 nM T67849 C7FDL2 71270817 IC50 = 15.85 nM T67849 CNR1G9 71270824 IC50 = 125.89 nM T67849 C38LBA 71270831 IC50 = 25.12 nM T67849 CTL6R5 71270836 IC50 = 19.95 nM T67849 CM4LX7 71270848 IC50 > 630.96 nM T67849 C2GWX6 71270906 IC50 > 501.19 nM T67849 CX0DL3 71270910 IC50 = 630.96 nM T67849 C0COW6 71270913 IC50 > 630.96 nM T67849 CB0S8G 71270927 IC50 = 6.31 nM T67849 C24IOW 71270948 IC50 > 630.96 nM T67849 C5BJ2Y 71270957 IC50 > 251.19 nM T67849 C03NFY 71271625 IC50 > 630.96 nM T67849 CL47JU 71271739 IC50 > 398.11 nM T67849 CS5JG6 71271910 IC50 = 100 nM T67849 C4PSK8 71271965 IC50 = 100 nM T67849 CB4N1M 71272066 IC50 > 630.96 nM T67849 CD8E1Y 71272453 IC50 = 25.12 nM T67849 C8EW9V 71272757 IC50 = 158.49 nM T67849 C0LO8I 71272765 IC50 = 79.43 nM T67849 C5A8WF 71449463 IC50 = 4 nM T67849 CWMY48 71450782 IC50 = 111 nM T67849 CNHJ63 71451228 IC50 = 8359 nM T67849 C7V3SO 71452608 IC50 = 139 nM T67849 C6KP3Z 71452609 IC50 < 600 nM T67849 C6W7ZU 71453081 IC50 = 0.6 nM T67849 CR84JX 71453419 Ki = 3 nM T67849 CZQW69 71453554 IC50 > 1000 nM T67849 CZ61FJ 71454160 IC50 = 31622776.6 nM T67849 CZ8Q5P 71454238 Ki = 1.2 nM T67849 C8QIB3 71454374 IC50 = 6 nM T67849 CGD6P2 71456119 IC50 = 3 nM T67849 CYR4J3 71456120 Ki = 3 nM T67849 CYL1G5 71456121 IC50 < 100 nM T67849 CG3OF4 71456597 IC50 = 1.9 nM T67849 CGL8Y4 71457063 IC50 = 6 nM T67849 CDG92F 71457924 IC50 = 14 nM T67849 CPI9J7 71457925 IC50 = 13 nM T67849 C9TAF0 71457926 IC50 = 40 nM T67849 CR14QX 71461548 IC50 = 260 nM T67849 CA6QB4 71461549 IC50 < 100 nM T67849 C3P4RX 71461550 IC50 < 200 nM T67849 CGE64P 71466531 IC50 = 210 nM T67849 CIHT92 71508937 IC50 = 120 nM T67849 CU3EO6 71520393 IC50 = 110 nM T67849 CYC6S1 71520394 IC50 = 2770 nM T67849 C1KMX0 71520395 IC50 = 458 nM T67849 CYK7N8 71520396 IC50 = 1120 nM T67849 CTC0O8 71520397 IC50 = 423 nM T67849 C0UZ3D 71526877 IC50 = 70 nM T67849 CP05SQ 71526878 IC50 = 2200 nM T67849 CZK6X9 71526879 IC50 = 3600 nM T67849 C8QRE4 71526880 IC50 = 1000 nM T67849 CT3QI8 71526881 IC50 = 1200 nM T67849 CO4MY1 71527005 IC50 = 390 nM T67849 CJC64F 71527006 IC50 = 670 nM T67849 C96WZG 71527007 IC50 = 58 nM T67849 CUC7I1 71527008 IC50 = 290 nM T67849 C09WKC 71527009 IC50 = 330 nM T67849 CSPO76 71527716 IC50 > 630.96 nM T67849 CIN7O1 71527842 IC50 > 630.96 nM T67849 CO6CI7 71528725 IC50 = 110 nM T67849 C5U2ZC 71528726 IC50 = 26 nM T67849 CTKO36 71528727 IC50 = 490 nM T67849 C2KF3X 71533728 IC50 = 152 nM T67849 CI7Q4K 71548718 IC50 = 28 nM T67849 CED62L 71548719 IC50 = 27 nM T67849 C4B0KN 71549093 IC50 = 720 nM T67849 C6PRV1 71655831 IC50 = 0.8 nM T67849 CF7R0Y 71682057 IC50 = 11000 nM T67849 CWG8M3 71682651 IC50 = 380 nM T67849 C6UGW3 71682652 IC50 = 4200 nM T67849 C7BX4K 71682653 IC50 = 770 nM T67849 CQX8N3 71682654 IC50 = 3300 nM T67849 CCG6J1 71682807 IC50 > 10000 nM T67849 CS32HB 71716798 IC50 = 251.19 nM T67849 C07GCV 71716799 IC50 > 630.96 nM T67849 CFW01E 71718034 IC50 = 128 nM T67849 C6XKV1 71819134 Ki = 2.3 nM T67849 C95VEJ 71819543 Ki = 0.59 nM T67849 CC3SY4 71819544 Ki = 0.9 nM T67849 CH5R0B 71819545 Ki = 0.88 nM T67849 C7EY1Q 72163951 Ki = 160 nM T67849 CVT76M 72163952 Ki = 490 nM T67849 C9UOH5 72164062 Ki > 10000 nM T67849 CT3X8G 72164184 Ki > 10000 nM T67849 CNX76A 72544842 IC50 = 1258.93 nM T67849 C29KOU 72709209 IC50 > 10000 nM T67849 CT73IW 72709284 IC50 > 10000 nM T67849 C9P1IG 72943510 IC50 = 2841 nM T67849 CVU2J9 72949025 IC50 = 2 nM T67849 CC6KY3 72949203 IC50 = 1 nM T67849 CYGV85 73051332 IC50 = 21 nM T67849 CV4BH5 73051810 IC50 = 21 nM T67849 C7N0AF 73052137 IC50 = 3 nM T67849 CNTD65 73052455 IC50 = 3 nM T67849 C8EI1X 73673707 IC50 = 3.8 nM T67849 CH75QS 73774946 IC50 = 4.4 nM T67849 CBYN18 73977439 IC50 = 15849 nM T67849 C9V1YR 73977449 IC50 = 2512 nM T67849 CXA90D 73977451 IC50 = 2512 nM T67849 CEZ7L2 73977461 IC50 = 794 nM T67849 CD0T9V 74539799 IC50 = 2.8 nM T67849 C16KOS 74539862 IC50 = 3.4 nM T67849 CQ0UM6 74763795 IC50 = 2210 nM T67849 CS71HC 74763798 IC50 = 2770 nM T67849 C5J4EC 76072924 IC50 = 3 nM T67849 CB7Z1L 76285656 EC50 = 1 nM T67849 C38UYZ 76286219 IC50 < 100 nM T67849 CN2MI8 76310247 IC50 > 50000 nM T67849 CKO41J 76310248 IC50 = 367 nM T67849 CEN9Q5 76310249 IC50 = 7600 nM T67849 CJCF67 76310250 IC50 = 14 nM T67849 CIBQ59 76311315 IC50 = 240 nM T67849 C8BD3K 76311316 IC50 = 90 nM T67849 C6F1CR 76311317 IC50 = 440 nM T67849 C7IDU0 76311318 IC50 = 640 nM T67849 CG40TB 76311319 IC50 > 1000 nM T67849 C5WSZ8 76311320 IC50 > 1000 nM T67849 C0M5SE 76311321 IC50 > 1000 nM T67849 CMR07I 76313939 IC50 > 50000 nM T67849 C5P2CJ 76313940 IC50 = 1140 nM T67849 CAV5Q9 76313941 IC50 = 836 nM T67849 CCY5L6 76314906 IC50 > 1000 nM T67849 CE3Z1I 76314907 IC50 = 1550 nM T67849 CFY10G 76314908 IC50 > 1000 nM T67849 C4UHR5 76314909 IC50 = 250 nM T67849 C1B3VO 76314910 IC50 > 1000 nM T67849 CY0Z4U 76314911 IC50 > 1000 nM T67849 CTVO82 76314912 IC50 > 1000 nM T67849 CCWP56 76314913 IC50 > 1000 nM T67849 C0J6PL 76317466 IC50 > 50000 nM T67849 CVW35P 76317467 IC50 > 50000 nM T67849 CZ1T3C 76317468 IC50 > 50000 nM T67849 C4MKN3 76317469 IC50 = 104 nM T67849 C3JA4F 76317470 IC50 = 770 nM T67849 C4XJ5Y 76317471 IC50 = 565 nM T67849 C3SIE7 76318525 IC50 > 1000 nM T67849 CU6G7L 76318526 IC50 > 1000 nM T67849 CC3Z2U 76318527 IC50 = 2000 nM T67849 C8E4GI 76321204 IC50 = 24 nM T67849 CF4OI8 76321205 IC50 = 1900 nM T67849 CR61ZP 76322185 IC50 > 1000 nM T67849 C5LT0B 76322186 IC50 > 1000 nM T67849 C19SKA 76322187 IC50 > 1000 nM T67849 CDG8V4 76324821 IC50 = 8 nM T67849 CJW39V 76324822 IC50 > 50000 nM T67849 C2BFA1 76324823 IC50 = 18 nM T67849 C1HFI9 76325446 IC50 = 430 nM T67849 C7IFD5 76325803 IC50 > 1000 nM T67849 C2NK4S 76325804 IC50 > 1000 nM T67849 COJ6P9 76325805 IC50 > 1000 nM T67849 C2AJ6T 76325806 IC50 > 1000 nM T67849 C4A8XZ 76328376 IC50 = 5280 nM T67849 C8S2IL 76329389 IC50 > 1000 nM T67849 CAEW42 76329390 IC50 > 1000 nM T67849 CMC32D 76329391 IC50 > 1000 nM T67849 CAZ9Q2 76329392 IC50 > 1000 nM T67849 C06ZQJ 76329393 IC50 = 3350 nM T67849 CYR0G6 76332050 IC50 = 150 nM T67849 C4MID5 76332051 IC50 = 26500 nM T67849 C70WJE 76332052 IC50 = 134 nM T67849 CE6BI0 76332666 IC50 = 63 nM T67849 CKG1E0 76333034 IC50 = 200 nM T67849 C6D4RU 76333035 IC50 > 1000 nM T67849 CSAT72 76333036 IC50 > 1000 nM T67849 C1JRO2 76333037 IC50 > 1000 nM T67849 C8TNI0 76333038 IC50 > 1000 nM T67849 C69ATM 76335666 IC50 > 50000 nM T67849 C0SI4C 76335667 IC50 > 50000 nM T67849 C31NEK 76335668 IC50 = 687 nM T67849 CL6BV5 76335669 IC50 = 11130 nM T67849 C73KJD 76335670 IC50 = 77 nM T67849 CP2UC5 76336660 IC50 > 1000 nM T67849 C79JAI 76336661 IC50 = 150 nM T67849 C2JTH8 77107528 IC50 = 1.9 nM T67849 C42HDP 77107927 IC50 = 4.1 nM T67849 C04SRC 77147259 IC50 = 3225 nM T67849 C9I7TY 78319187 IC50 = 12589.25 nM T67849 C24LQH 78320362 IC50 = 4 nM T67849 C9T8KF 78320671 IC50 < 3 nM T67849 CI2YN8 78320672 IC50 < 3 nM T67849 CI6K4J 78320673 IC50 = 52 nM T67849 COFJ16 78320996 IC50 = 76 nM T67849 CMU5P2 78321310 IC50 = 14 nM T67849 CE13AJ 78321314 IC50 = 11 nM T67849 CSP2H4 78321635 IC50 = 8 nM T67849 CWA0B1 78322567 IC50 = 12 nM T67849 CH6P9D 78322877 IC50 = 43 nM T67849 C4IW9V 78323193 IC50 = 23 nM T67849 CD1JC8 78324443 IC50 = 5 nM T67849 C04IKP 86268622 IC50 = 2.5 nM T67849 C5P3RO 86647783 IC50 = 620 nM T67849 CP7HJ2 86666761 IC50 = 99 nM T67849 CD6XP5 86677746 IC50 = 11 nM T67849 CDXM47 86677874 IC50 < 1 nM T67849 CP3W1B 86695297 IC50 = 15 nM T67849 CA17UE 86732669 IC50 = 9 nM T67849 C2PCS7 87061302 IC50 = 223 nM T67849 CI8X3C 87150169 IC50 = 12589.25 nM T67849 CV6PI8 87562294 IC50 = 316.23 nM T67849 CN4B6P 88536250 IC50 = 5.3 nM T67849 C1HB3F 89051931 IC50 = 8.2 nM T67849 CY64GN 89420800 IC50 = 1.9 nM T67849 C61SCX 89493851 IC50 = 4.9 nM T67849 C1LU3X 89493904 IC50 = 29 nM T67849 CTE1L0 89517065 IC50 = 9 nM T67849 C56KSC 89517226 IC50 = 36 nM T67849 CN5Y9A 90064110 IC50 = 16 nM T67849 C7FP2M 90064111 IC50 = 5 nM T67849 CQE9C3 90158083 IC50 = 8330 nM T67849 C9IOQ0 90158408 IC50 = 45 nM T67849 C9JAI2 90166620 IC50 = 572 nM T67849 C49XDA 90166847 IC50 = 190 nM T67849 CC4M6F 90168602 IC50 = 35 nM T67849 C5LK7G 90168751 IC50 = 1290 nM T67849 CF03DW 90168772 IC50 = 24 nM T67849 CM6J9K 90168778 IC50 = 16 nM T67849 CVF37R 90168935 IC50 = 187 nM T67849 C28WQY 90431726 IC50 = 30 nM T67849 C08UWK 90665816 IC50 = 630 nM T67849 CMWB58 91757958 IC50 <= 10000 nM T67849 C3Y0DS 91801158 IC50 = 59 nM T67849 C2OG7F 91820679 IC50 = 0.7 nM T67849 CAS7W6 91864650 IC50 = 880 nM T67849 C1QJ3K 117815397 IC50 = 4200 nM T67849 CLA03N 117965586 IC50 = 2 nM T67849 C34FKB 118025462 IC50 = 4 nM T67849 CUQS80 118025552 IC50 = 13 nM T67849 C1KGB4 118025559 IC50 = 1830 nM T67849 CDF6L7 118025606 IC50 = 1340 nM T67849 CGX1T6 118025676 IC50 = 61 nM T67849 C1IL8Q 118025680 IC50 = 9 nM T67849 C79ZBM 118025723 IC50 = 33 nM T67849 C6HO9P 118025760 IC50 = 8 nM T67849 CM4Z5V 118025790 IC50 = 2790 nM T67849 CX4W9A 118025823 IC50 = 35 nM T67849 C3FG4U 118025830 IC50 = 32 nM T67849 CM3JO2 118025835 IC50 = 155 nM T67849 CKR9G1 118025928 IC50 = 3 nM T67849 C5TQU3 118025943 IC50 = 8 nM T67849 C68YAU 118026010 IC50 = 172 nM T67849 C14WCU 118131317 IC50 < 10 nM T67849 CE42ID 118165924 IC50 = 0.04 nM T67849 C67VQE 118341819 IC50 > 10000 nM T67849 CC9P5H 118341835 IC50 > 10000 nM T67849 CUMA23 118341844 IC50 = 270 nM T67849 C3IP9X 118341852 IC50 > 10000 nM T67849 C6TI0Z 118341865 IC50 > 10000 nM T67849 C4U7NC 118341870 IC50 > 10000 nM T67849 CVL03K 118341884 IC50 > 10000 nM T67849 CPZN96 118341923 IC50 > 10000 nM T67849 C9E3DU 118341927 IC50 > 10000 nM T67849 CVN87P 118433737 IC50 = 2.7 nM T67849 C8W1RN 118445922 IC50 = 3 nM T67849 CQF1V4 118446049 IC50 = 63 nM T67849 CVYK24 118556943 IC50 = 62 nM T67849 CJQ92T 118572891 IC50 = 10 nM T67849 C2U3BQ 118627731 IC50 = 0.1 nM T67849 CS5C8W 118684133 IC50 = 4.1 nM T67849 CRX24W 118709077 IC50 = 110 nM T67849 CV2EJ7 118709081 IC50 = 85 nM T67849 CZ41AQ 118709092 IC50 = 400 nM T67849 CR6ML1 118709578 IC50 = 51 nM T67849 C0OH7I 118709579 IC50 = 230 nM T67849 C73YIO 118709582 IC50 = 45 nM T67849 CGWX02 118709583 IC50 = 32 nM T67849 CB53EU 118728320 IC50 > 50000 nM T67849 C6KJL1 118728321 IC50 = 42618 nM T67849 CKJ3S6 118728322 IC50 > 50000 nM T67849 CT0L3Y 118728325 IC50 > 50000 nM T67849 CHS2E4 118728326 IC50 > 50000 nM T67849 CRUP47 118728328 IC50 = 47763 nM T67849 CQR41G 118728330 IC50 = 39842 nM T67849 CN4Q9R 118728332 IC50 = 34624 nM T67849 CDI10F 118728336 IC50 > 50000 nM T67849 CHT6K9 118728811 Ki > 4000 nM T67849 CUA3Y2 118728812 Ki > 4000 nM T67849 CDQ78G 118728813 Ki = 3100 nM T67849 CZ6XL7 118728814 Ki = 180 nM T67849 CMO67K 118728815 Ki > 4000 nM T67849 CR2M0Q 118728816 Ki > 4000 nM T67849 C62SCL 118728817 Ki > 4000 nM T67849 CSB30C 118728819 Ki = 1900 nM T67849 CV7XU8 118728820 Ki = 1600 nM T67849 C3J1EX 118728821 Ki > 4000 nM T67849 CIWB78 118728822 Ki > 4000 nM T67849 CP18SE 118728823 Ki > 4000 nM T67849 CM42CA 118728824 Ki = 2500 nM T67849 C9Q7CL 118728825 Ki = 1200 nM T67849 CCR3S0 118728826 Ki = 3300 nM T67849 CB1WC5 118729946 IC50 = 2.5 nM T67849 CQ4G9M 118729947 IC50 = 1.7 nM T67849 C43IPJ 118729948 IC50 = 4 nM T67849 C3I9CQ 118729949 IC50 = 1.4 nM T67849 CZQ17M 118729950 IC50 = 1.2 nM T67849 C3G1ZP 118729951 IC50 = 3.1 nM T67849 CY60FC 118730033 IC50 > 50000 nM T67849 CN3B4U 118730711 IC50 = 22 nM T67849 C0IL3N 118730712 IC50 = 23 nM T67849 C3CH1A 118730713 IC50 = 20 nM T67849 CHX5L9 118730714 IC50 = 14 nM T67849 CNJ32C 118730715 IC50 = 80 nM T67849 C1MKB3 118730716 IC50 = 27 nM T67849 C81RJA 118730717 IC50 = 160 nM T67849 CFZ16R 118737301 IC50 <= 10000 nM T67849 C27CPQ 118737302 IC50 <= 10000 nM T67849 C59VXA 118737303 IC50 <= 10000 nM T67849 CGO1N4 118737304 IC50 <= 10000 nM T67849 CS85FM 118737305 IC50 <= 10000 nM T67849 C8UCO1 118737306 IC50 <= 10000 nM T67849 CR0BZ2 118737307 IC50 <= 10000 nM T67849 C3N4DJ 118737308 IC50 <= 10000 nM T67849 CGY5B1 118737309 IC50 <= 10000 nM T67849 CFN12W 121445751 IC50 = 25.8 nM T67849 CVU7P1 121445752 IC50 = 0.6 nM T67849 C2UDS6 121445784 IC50 = 6 nM T67849 C04NDW 121445810 IC50 = 17.4 nM T67849 CM4Y3Z 121483558 IC50 = 309 nM T67849 C81IFQ 122163152 IC50 = 1840 nM T67849 C2VGD5 122178120 IC50 = 13.3 nM T67849 C24XUZ 122178124 IC50 = 3.1 nM T67849 CN5AB3 122179486 IC50 = 10 nM T67849 CLEK13 122179487 IC50 = 4 nM T67849 C0OW8H 122179490 IC50 = 44 nM T67849 C0VD5F 122179491 IC50 = 63.1 nM T67849 CQ87FB 122179492 IC50 = 199 nM T67849 CBJ29X 122179493 IC50 = 2000 nM T67849 CA5N1B 122179494 IC50 = 20 nM T67849 CSTE64 122179689 IC50 = 220 nM T67849 CE2FM7 122179690 IC50 = 470 nM T67849 CZJ31R 122179691 IC50 = 270 nM T67849 CBOU30 122179692 IC50 = 470 nM T67849 CKWC74 122179693 IC50 = 810 nM T67849 C4CX7Z 122179694 IC50 = 710 nM T67849 C48LYC 122179695 IC50 = 1100 nM T67849 C3D5QM 122179696 IC50 = 240 nM T67849 CW3DM7 122179697 IC50 = 600 nM T67849 C6I3PB 122179698 IC50 > 10000 nM T67849 CCU6A4 122179699 IC50 = 570 nM T67849 C7WMC3 122179700 IC50 = 470 nM T67849 C86NOQ 122179701 IC50 = 550 nM T67849 CAHY19 122179702 IC50 = 460 nM T67849 C3O7CM 122179703 IC50 = 1500 nM T67849 CK2R4X 122179704 IC50 = 410 nM T67849 CG96HD 122179705 IC50 = 900 nM T67849 C1PK9L 122179706 IC50 = 470 nM T67849 CEB69W 122179707 IC50 = 1000 nM T67849 CK97EL 122179708 IC50 = 500 nM T67849 C0ZA4C 122179709 IC50 = 640 nM T67849 CU93YJ 122179710 IC50 = 450 nM T67849 C0KTH8 122179711 IC50 = 150 nM T67849 CN9I1C 122179712 IC50 = 530 nM T67849 C65OGI 122179713 IC50 = 300 nM T67849 C92AZK 122179714 IC50 = 140 nM T67849 CWL43Z 122179715 IC50 > 10000 nM T67849 C50VNH 122179716 IC50 > 10000 nM T67849 COW37C 122179717 IC50 > 10000 nM T67849 CG5N9E 122179718 IC50 = 220 nM T67849 CB14FW 122179719 IC50 = 270 nM T67849 CHZ3S1 122179720 IC50 = 470 nM T67849 CEG8Y6 122179721 IC50 = 30 nM T67849 CG5P3J 122179722 IC50 = 1700 nM T67849 CZH3T1 122179723 IC50 = 480 nM T67849 C10FGR 122179724 IC50 = 1800 nM T67849 CEFS13 122180793 IC50 = 14570 nM T67849 CFZ2E1 122180794 IC50 = 20120 nM T67849 C5YKG7 122180795 IC50 = 71350 nM T67849 C9ID7U 122180796 IC50 = 56890 nM T67849 C08XOC 122180839 IC50 = 120000 nM T67849 C2HM6P 122180840 IC50 = 154780 nM T67849 CT9Y6U 122180841 IC50 = 3550 nM T67849 C6FOM0 122180842 IC50 = 2740 nM T67849 COX90L 122180843 IC50 = 1810 nM T67849 CP40RU 122180844 IC50 = 3970 nM T67849 CC0EK9 122180845 IC50 = 2610 nM T67849 CS85CU 122181413 IC50 = 20 nM T67849 CQS67B 122181416 IC50 = 17 nM T67849 C58XRY 122184465 IC50 = 3981.07 nM T67849 C16ALM 122184466 IC50 = 1995.26 nM T67849 CIX19J 122184467 IC50 = 6309.57 nM T67849 CDZY02 122184468 IC50 = 63095.73 nM T67849 CTH70U 122184469 IC50 = 12589.25 nM T67849 C9ZXR7 122184470 IC50 = 6309.57 nM T67849 CNJ9Z4 122184471 IC50 = 12589.25 nM T67849 CS41EG 122184473 IC50 = 1258.93 nM T67849 CZ36GL 122184474 IC50 = 1000 nM T67849 CU4ZT6 122184475 IC50 = 12589.25 nM T67849 C3H9PR 122184476 IC50 = 1995.26 nM T67849 CU40TW 122184477 IC50 = 6309.57 nM T67849 CAMD31 122184479 IC50 = 63095.73 nM T67849 C1F9RK 122184480 IC50 = 1258.93 nM T67849 C7XW1K 122184481 IC50 = 79432.82 nM T67849 CRUX54 122184482 IC50 = 50118.72 nM T67849 CQ7W0P 122184526 IC50 = 7943.28 nM T67849 CA5YB2 122184529 IC50 = 12589.25 nM T67849 C64YPH 122184530 IC50 = 25118.86 nM T67849 C4AGX5 122184531 IC50 = 19952.62 nM T67849 CQL4K5 122184532 IC50 = 12589.25 nM T67849 CRKV74 122184533 IC50 = 19952.62 nM T67849 CX14YD 122184534 IC50 = 3981.07 nM T67849 CM6A4S 122184535 IC50 = 19952.62 nM T67849 CF86YS 122184536 IC50 = 19952.62 nM T67849 CH08SN 122184537 IC50 = 5011.87 nM T67849 CYRH97 122184538 IC50 = 10000 nM T67849 CD4W0Z 122184539 IC50 > 199526.23 nM T67849 CH8Y3Q 122184540 IC50 = 100000 nM T67849 CDA85R 122184541 IC50 > 199526.23 nM T67849 CF36XJ 122184542 IC50 > 199526.23 nM T67849 CQ6O7H 122184543 IC50 > 199526.23 nM T67849 CS4MN0 122184544 IC50 > 79432.82 nM T67849 CKT74G 122185265 IC50 = 16 nM T67849 CJ6C1O 122185267 IC50 = 12 nM T67849 CK9VY5 122197304 IC50 < 50 nM T67849 CGW35U 122387497 IC50 > 1000 nM T67849 C38BML 122387499 IC50 > 1000 nM T67849 CCW0M1 122387500 IC50 = 553 nM T67849 CKA90Y 122387501 IC50 = 348 nM T67849 CH4LC6 122387502 IC50 = 271 nM T67849 C8OC3E 122387504 IC50 = 674 nM T67849 C34AHY 122387505 IC50 = 722 nM T67849 CUG1T6 122387506 IC50 = 311 nM T67849 CE7K5C 122387507 IC50 = 683 nM T67849 C4HL3N 122387508 IC50 = 474 nM T67849 CA7L3S 122387509 IC50 = 489 nM T67849 CR9NF3 122542400 IC50 = 1.4 nM T67849 CMG21L 122705987 IC50 = 8500 nM T67849 CW5EK9 122705988 IC50 = 640 nM T67849 CPTY78 124518210 IC50 = 2.5 nM T67849 C1N6YP 126480569 IC50 = 110 nM T67849 CE52HC 126480570 IC50 = 90 nM T67849 CPW54V 126480574 IC50 = 50 nM T67849 CVJ3Q5 127025094 IC50 > 1000 nM T67849 C98DKI 127025346 IC50 = 19 nM T67849 CBXJ67 127025628 IC50 = 14 nM T67849 CSV3R7 127029064 IC50 = 50 nM T67849 CQTG79 127029604 IC50 > 1000 nM T67849 C47BCU 127030580 IC50 = 740 nM T67849 CZHT45 127031017 IC50 = 1570 nM T67849 CU0F4R 127031332 IC50 = 340 nM T67849 C2IN4Q 127031333 IC50 = 50000 nM T67849 CS12RU 127031435 IC50 = 12.4 nM T67849 CGU4H3 127031891 IC50 = 33 nM T67849 CGKR53 127032915 IC50 = 2075 nM T67849 CYSN74 127034047 IC50 = 3700 nM T67849 C41YQI 127035981 IC50 > 5000 nM T67849 C2O4RK 127038523 IC50 = 2600 nM T67849 CO27IE 127038894 IC50 = 10000 nM T67849 C72NPR 127039226 IC50 = 4500 nM T67849 CL0ZU8 127040691 IC50 = 2700 nM T67849 CB0G7Z 127040692 IC50 = 10000 nM T67849 C3ZXT2 127040693 IC50 = 9000 nM T67849 CY6NM3 127040694 IC50 > 10000 nM T67849 CLUK47 127042289 IC50 = 12000 nM T67849 C05MRE 127042767 IC50 = 4800 nM T67849 C4L9TC 127042949 IC50 = 3700 nM T67849 CG8DA9 127045861 IC50 = 505 nM T67849 CVF8Z9 127045862 IC50 = 7.3 nM T67849 CH68NT 127046076 IC50 = 149 nM T67849 CA2XD5 127046077 IC50 = 221 nM T67849 COJ68G 127046117 IC50 = 13 nM T67849 C34REM 127046317 IC50 = 11 nM T67849 CC4ND8 127046862 IC50 = 271 nM T67849 CY2P1X 127047138 IC50 = 11 nM T67849 CZ2R0C 127047140 IC50 = 10 nM T67849 CT89GI 127047683 IC50 = 14 nM T67849 C7D0FN 127047685 IC50 = 7 nM T67849 CN94CQ 127047797 IC50 = 9 nM T67849 C5OE2H 127053611 IC50 = 71 nM T67849 CN9XL1 129262531 IC50 = 1 nM T67849 C92EMK 129395626 IC50 = 3.6 nM T67849 CW7A5X 129626595 IC50 = 31.62 nM T67849 CGIT40 129896911 IC50 = 16 nM T67849 C18NHD 130302549 IC50 <= 10000 nM T67849 CL13RZ 130302558 IC50 <= 10000 nM T67849 CF5JZ3 130302563 IC50 <= 10000 nM T67849 CD46EL 130302605 IC50 <= 10000 nM T67849 CNI8M6 130302620 IC50 <= 10000 nM T67849 CI6WN9 130302651 IC50 <= 10000 nM T67849 C5ZP0L 130302658 IC50 <= 10000 nM T67849 CW61SG 130302663 IC50 <= 10000 nM T67849 CB27ZG 130302668 IC50 <= 10000 nM T67849 C5VYM6 130302674 IC50 <= 10000 nM T67849 C0FQR2 130302675 IC50 <= 10000 nM T67849 CB34HQ 130302676 IC50 <= 10000 nM T67849 CQR1I8 130302685 IC50 <= 10000 nM T67849 C17DZF 130302698 IC50 <= 10000 nM T67849 CBC6W7 130302701 IC50 <= 10000 nM T67849 CBT21G 130302702 IC50 <= 10000 nM T67849 CDZ45O 130302703 IC50 <= 10000 nM T67849 C2GWU8 130302709 IC50 <= 10000 nM T67849 CV3M6Y 130302710 IC50 <= 10000 nM T67849 C39UQN 130302731 IC50 <= 10000 nM T67849 CL9O8X 130302732 IC50 <= 10000 nM T67849 CL69GM 130302740 IC50 <= 10000 nM T67849 CH8YK9 130302741 IC50 <= 10000 nM T67849 CQR2W9 130302781 IC50 <= 10000 nM T67849 C9HC8A 130302803 IC50 <= 10000 nM T67849 CIK25W 130302809 IC50 <= 10000 nM T67849 CI08PF 130332501 IC50 <= 10000 nM T67849 C1H4UT 130332505 IC50 <= 10000 nM T67849 CZPI64 130332579 IC50 <= 10000 nM T67849 CDS9F3 130332582 IC50 <= 10000 nM T67849 C3G0HF 130332585 IC50 <= 10000 nM T67849 CX13UC 130332620 IC50 <= 10000 nM T67849 CED6F3 130332657 IC50 <= 10000 nM T67849 CRG3I4 130362847 IC50 = 0.8 nM T67849 C8W2EJ 130362892 IC50 = 5.2 nM T67849 C3YFV8 130362899 IC50 = 1.8 nM T67849 CP5D7R 130362915 IC50 = 0.4 nM T67849 CUP5N0 130363024 IC50 = 0.6 nM T67849 CD1PV2 130363056 IC50 = 3.5 nM T67849 CKTL52 130363065 IC50 = 2.5 nM T67849 CR8S9K 130363066 IC50 = 5 nM T67849 CJ3Y7M 130363067 IC50 = 7 nM T67849 C19CXK 130363082 IC50 = 1.2 nM T67849 COS6W5 130363083 IC50 = 56 nM T67849 CO1YL7 130363101 IC50 = 24 nM T67849 CE1YZ2 130363102 IC50 = 2.4 nM T67849 CBN3D6 130363112 IC50 = 1 nM T67849 C3QBL4 130363125 IC50 = 0.3 nM T67849 C53JWU 130363129 IC50 = 1.9 nM T67849 C3SK4J 130363145 IC50 = 72 nM T67849 CX8D6O 130363152 IC50 = 3 nM T67849 CK91CJ 130363160 IC50 = 105 nM T67849 C0A2YT 130363168 IC50 = 1 nM T67849 C7E6XI 130363172 IC50 = 0.5 nM T67849 C7JP0R 130363201 IC50 = 3.3 nM T67849 C76YRN 130363211 IC50 = 3 nM T67849 C3Q7LT 130363215 IC50 = 0.9 nM T67849 C7OPB5 130363224 IC50 = 1.9 nM T67849 C64XBS 130363239 IC50 = 98 nM T67849 CN75CD 130363275 IC50 = 4.8 nM T67849 CYTF09 130363280 IC50 = 31 nM T67849 CLAB53 130363290 IC50 = 140 nM T67849 CFI60X 130363298 IC50 = 1.1 nM T67849 C3V9DW 130363308 IC50 > 150 nM T67849 CNO3U9 130363327 IC50 = 5 nM T67849 COKX96 130363382 IC50 = 1 nM T67849 CJO36T 130363391 IC50 = 2 nM T67849 CFXC13 130363397 IC50 = 0.4 nM T67849 C0WS3I 130363410 IC50 = 9 nM T67849 C60KGA 130363411 IC50 = 1.1 nM T67849 C31RSQ 130363418 IC50 = 2 nM T67849 CTN8C0 130363443 IC50 = 1.4 nM T67849 CD54NU 130363457 IC50 = 5 nM T67849 C3PB1V 130363463 IC50 = 4 nM T67849 CNFH51 130363544 IC50 = 0.8 nM T67849 C65ZDT 130363548 IC50 = 5 nM T67849 CULX27 130363568 IC50 = 30 nM T67849 COK9T6 130363592 IC50 = 33 nM T67849 C6CIJ2 130363602 IC50 = 1.5 nM T67849 CFN3Z5 130363612 IC50 = 6 nM T67849 CMX9O5 130363616 IC50 = 5.5 nM T67849 C6H9BS 130363645 IC50 = 2.1 nM T67849 COPI97 130363656 IC50 = 5.5 nM T67849 C0G9LM 130363659 IC50 = 2 nM T67849 COWE45 130363737 IC50 < 0.3 nM T67849 CAK3T1 130363738 IC50 = 2 nM T67849 CR8G9C 130363746 IC50 = 2 nM T67849 C47CAY 130421765 IC50 = 794.33 nM T67849 C84YKI 130422161 IC50 = 398.11 nM T67849 CK68CA 130453737 IC50 = 730 nM T67849 CDE7T3 132005217 IC50 = 120 nM T67849 CL26YS 132005219 IC50 = 96 nM T67849 CP32GB 132005220 IC50 = 29 nM T67849 CG1NC4 132005221 IC50 = 2600 nM T67849 C0UV2M 132005224 IC50 = 41 nM T67849 CUN18W 132005225 IC50 = 2 nM T67849 CD84OI 132005228 IC50 = 1.5 nM T67849 C9VDI0 132005229 IC50 = 230 nM T67849 CB1Z7P 132005231 IC50 = 440 nM T67849 C7ASP9 132005246 IC50 = 1.7 nM T67849 C8VE6T 132005248 IC50 = 51 nM T67849 C7LCW1 132005249 IC50 = 76 nM T67849 C5W9LN 132005323 IC50 = 20 nM T67849 CQ6GO2 132005326 IC50 = 39 nM T67849 C1XUW7 132209432 IC50 = 4.7 nM T67849 CPL60M 132209468 IC50 = 0.6 nM T67849 C6Y4CH 132209868 IC50 = 4 nM T67849 C58NEJ 132209870 IC50 = 19 nM T67849 CIL1Q3 132209885 IC50 = 6.4 nM T67849 CP7N3I 132209920 IC50 = 3 nM T67849 C4M8WN 132209922 IC50 = 1.3 nM T67849 CJ83PK 132209926 IC50 = 3.9 nM T67849 CJ5FI1 132209935 IC50 = 11 nM T67849 CHQP87 132209952 IC50 = 100 nM T67849 C6JGE1 132209957 IC50 = 1.7 nM T67849 C45NEF 132209959 IC50 = 5.5 nM T67849 CZFO16 132209976 IC50 = 1.2 nM T67849 CI6P5H 132209981 IC50 = 6 nM T67849 CCK6E1 132209985 IC50 = 10 nM T67849 COK4X3 132210002 IC50 = 0.9 nM T67849 CTG6C8 132210009 IC50 = 2 nM T67849 C3CFB2 132210012 IC50 = 4.5 nM T67849 CS4V6U 132210025 IC50 = 0.9 nM T67849 CM9P1H 132210051 IC50 = 424 nM T67849 C16HBK 132210068 IC50 = 1.3 nM T67849 CFI23B 132210082 IC50 = 0.5 nM T67849 C02QSJ 132210090 IC50 = 16 nM T67849 C9Q0ZW 132210105 IC50 = 16 nM T67849 CH8DP7 132220479 IC50 < 0.1 nM T67849 C6NWY1 132220480 IC50 = 1 nM T67849 CD7X5S 132220481 IC50 = 2.2 nM T67849 CRC14V 132220484 IC50 = 1.5 nM T67849 C4Q5LF 132471857 IC50 = 7 nM T67849 CJE34F 132597748 IC50 = 18.5 nM T67849 CCV46G 132606879 IC50 = 3.981 nM T67849 C6PWX2 134129963 IC50 = 66 nM T67849 CV2PK1 134129977 IC50 = 100 nM T67849 CSWZ68 134130018 IC50 = 61 nM T67849 CBR3Z9 134130128 IC50 = 88 nM T67849 CM51SI 134130327 IC50 = 55 nM T67849 CLO3M4 134130336 IC50 = 470 nM T67849 CS9Q7P 134130420 IC50 = 575 nM T67849 C0WEA6 134130582 IC50 = 60 nM T67849 C2X1BY 134130678 IC50 = 150 nM T67849 C97JFV 134131108 IC50 = 68 nM T67849 C1LZP4 134131157 IC50 = 100 nM T67849 COI4W0 134131210 IC50 > 1000 nM T67849 C54IJX 134131348 IC50 = 170 nM T67849 C5M6BU 134131349 IC50 = 350 nM T67849 CH17GQ 134131392 IC50 = 130 nM T67849 CIYZ86 134131408 IC50 = 658 nM T67849 C9NYX3 134131539 IC50 = 370 nM T67849 CFG90E 134132909 IC50 = 256 nM T67849 CI49TK 134133218 IC50 = 1.6 nM T67849 C4YNH0 134134126 IC50 = 28 nM T67849 C0EK8P 134134680 IC50 = 11 nM T67849 CU9VC6 134136072 IC50 = 47 nM T67849 CS73WF 134136130 IC50 = 370 nM T67849 C0A1UM 134138053 IC50 = 10 nM T67849 C6OGM2 134138249 IC50 = 120 nM T67849 CQ2S4X 134138703 IC50 = 188 nM T67849 CQUY75 134139416 IC50 = 51 nM T67849 CL3Q6G 134140420 IC50 = 130 nM T67849 C0PN3R 134140590 IC50 = 55 nM T67849 CN5VU4 134142014 IC50 = 3.8 nM T67849 CDJ10M 134142931 IC50 = 146 nM T67849 CUE85S 134143151 IC50 = 5600 nM T67849 CN59WG 134143270 IC50 = 1090 nM T67849 CL4E9X 134144824 IC50 = 330 nM T67849 CQ9G7H 134145670 IC50 = 9 nM T67849 C1PVM6 134145863 IC50 = 9100 nM T67849 C6G8EJ 134146051 IC50 = 55000 nM T67849 CIPL93 134147099 IC50 = 110 nM T67849 C8ITR3 134147904 IC50 = 7700 nM T67849 CV2QA7 134148173 IC50 = 1000 nM T67849 CXA3V0 134148445 IC50 = 488 nM T67849 C3FO5C 134149163 IC50 = 740 nM T67849 CY3HC4 134150338 IC50 = 11 nM T67849 CXU92M 134150578 IC50 = 15 nM T67849 CG8LE2 134151667 IC50 < 10000 nM T67849 CK43EY 134152988 IC50 = 22 nM T67849 CL5MR8 134154147 IC50 = 17000 nM T67849 CS2QP7 134154582 IC50 = 16 nM T67849 C2QGB3 134156160 IC50 = 5 nM T67849 CV89ZY 134157127 IC50 = 16 nM T67849 C42RJH 134157534 IC50 = 9 nM T67849 C2SE0Y 134157628 IC50 = 0.2 nM T67849 CDSB36 134248984 IC50 = 0.6166 nM T67849 CKP8O2 134249145 Ki = 7800 nM T67849 CA3U2C 134519452 IC50 = 719 nM T67849 CEO8F9 134519632 IC50 = 106 nM T67849 CKH7O4 134519691 IC50 = 20 nM T67849 CTD03Q 134611885 IC50 = 1.259 nM T67849 CJXA12 134611894 IC50 = 1000 nM T67849 CWZ39C 134823450 IC50 = 1.4 nM T67849 C14AOZ 134823456 IC50 < 1 nM T67849 C54FXD 134957362 IC50 = 158.49 nM T67849 C9FUK2 135151360 IC50 > 30000 nM T67849 CT0GQ6 135197577 IC50 = 0.35 nM T67849 C87VKA 135197594 IC50 = 0.37 nM T67849 CQXS07 135197635 IC50 = 0.23 nM T67849 C7KXF1 135197643 IC50 = 0.18 nM T67849 CY38TL 135391000 IC50 = 2.8 nM T67849 COG86Z 135397763 IC50 = 125.89 nM T67849 CWL67T 135397764 IC50 = 6.31 nM T67849 CX8AI4 135398491 IC50 = 58 nM T67849 CH8TR5 135426721 IC50 = 4000 nM T67849 C7SND1 135429301 IC50 < 100 nM T67849 C6AZ2R 135435018 IC50 = 25118.86 nM T67849 C3QJ8W 135566371 IC50 = 9 nM T67849 C24ZGX 135566644 IC50 = 1395 nM T67849 C2QDV5 135566741 IC50 = 118 nM T67849 C2UN0D 135742360 IC50 = 6400 nM T67849 CU29YK 135750268 IC50 = 84 nM T67849 C02PHA 135927892 IC50 = 6309.57 nM T67849 CS8T3D 135927897 IC50 = 501.19 nM T67849 C12UDA 135947972 IC50 = 161 nM T67849 CN42ZS 135947973 IC50 = 250 nM T67849 CF8AO3 135947974 IC50 = 90 nM T67849 CW08GJ 135947976 IC50 = 66 nM T67849 C8O9HG 135947977 IC50 = 100000 nM T67849 CJN7E2 135947978 IC50 = 61 nM T67849 CFKH34 135947979 IC50 = 59 nM T67849 C0ZH9X 135981194 IC50 = 25560 nM T67849 C4G2HP 135995897 IC50 = 1680 nM T67849 CNF15Q 135995898 IC50 = 320 nM T67849 C98HZG 135995899 IC50 = 1020 nM T67849 CIQ82W 135995900 IC50 = 880 nM T67849 CD57NX 136027097 Ki = 2.85 nM T67849 CP1US5 136041737 IC50 = 164 nM T67849 CXH63V 136041747 IC50 = 219 nM T67849 C6B5TC 136041748 IC50 = 779 nM T67849 CU6XG1 136041749 IC50 = 442 nM T67849 C0U5DB 136041750 IC50 = 397 nM T67849 C48KAQ 136041752 IC50 = 9040 nM T67849 C74PRL 136041753 IC50 = 854 nM T67849 CT4FJ1 136041757 IC50 = 28 nM T67849 CCS2G6 136041761 IC50 = 1137 nM T67849 CEZP21 136041762 IC50 = 855 nM T67849 CJ58TD 136041764 IC50 = 2555 nM T67849 CX67QW 136041765 IC50 = 36 nM T67849 CK0H2Q 136041766 IC50 = 84 nM T67849 CQP7B6 136041767 IC50 = 3360 nM T67849 CM65BS 136041773 IC50 = 225 nM T67849 C6P7JB 136041775 IC50 = 247 nM T67849 C5CJF7 136041776 IC50 = 36 nM T67849 C3XIZ8 136041777 IC50 = 270 nM T67849 C32LKO 136041785 IC50 = 2210 nM T67849 C90ARP 136041787 IC50 = 2850 nM T67849 CZ3BN1 136041792 IC50 = 122 nM T67849 CG19DI 136041799 IC50 = 21 nM T67849 CXJA29 136041804 IC50 = 87 nM T67849 CHT31V 136041805 IC50 = 17 nM T67849 CO8C4J 136041817 IC50 = 6 nM T67849 C4QU6G 136041827 IC50 = 4135 nM T67849 CNE10X 136041834 IC50 = 648 nM T67849 CS3AE1 136041847 IC50 = 86 nM T67849 CZC47Y 136041848 IC50 = 278 nM T67849 CA91JG 136069599 IC50 = 18 nM T67849 CGAB91 136069600 IC50 = 34 nM T67849 C3ZAW2 136069605 IC50 = 98 nM T67849 C8JXL5 136069609 IC50 = 22 nM T67849 C9I0EQ 136069610 IC50 = 106 nM T67849 C25EYJ 136069611 IC50 = 7 nM T67849 C2S5QF 136069615 IC50 = 2 nM T67849 CC4UM3 136176116 IC50 = 180 nM T67849 CJRK81 136176117 IC50 = 274 nM T67849 C63IOS 136176118 IC50 = 181 nM T67849 C3KW7H 136176119 IC50 = 6748 nM T67849 C69AKQ 136176120 IC50 = 3406 nM T67849 CF17KO 136176121 IC50 = 8450 nM T67849 CU3TE0 136176122 IC50 = 2755 nM T67849 C3X5KE 136176124 IC50 = 2385 nM T67849 CA8C5E 136176125 IC50 = 2271 nM T67849 C5OMG2 136176126 IC50 = 373 nM T67849 CP2YM7 136176127 IC50 = 1181 nM T67849 C8XIJ0 136176128 IC50 = 398 nM T67849 CUY8N4 136176129 IC50 = 2170 nM T67849 C3J4ME 136176130 IC50 = 335 nM T67849 CR1NZ2 136176131 IC50 = 995 nM T67849 C4WG2F 136176132 IC50 = 151 nM T67849 CJ8EC5 136176139 IC50 = 1060 nM T67849 CQ84IZ 136180335 Ki > 4000 nM T67849 C1LK9U 136183381 IC50 = 55 nM T67849 C27TKQ 136196449 IC50 = 22 nM T67849 CK9S4X 136229137 IC50 = 140 nM T67849 C7S1YJ 136230225 IC50 = 2450 nM T67849 C3Q6ED 136230226 IC50 = 1108 nM T67849 CKPF02 136230227 IC50 = 4270 nM T67849 CZY9O0 136230228 IC50 = 2783 nM T67849 CRET01 136230229 IC50 = 611 nM T67849 CX1KI8 136230230 IC50 = 189 nM T67849 C3Z5MH 136230231 IC50 = 135 nM T67849 CUE6N8 136230232 IC50 = 63 nM T67849 C8Q1AP 136230233 IC50 = 137 nM T67849 C70RXE 136230234 IC50 = 148 nM T67849 C4W0KN 136230235 IC50 = 297 nM T67849 CMZN01 136230236 IC50 = 4647 nM T67849 CCU0H5 136241428 IC50 = 24 nM T67849 C4QMY7 136244246 IC50 = 11530 nM T67849 CF3DK1 136245085 IC50 = 24030 nM T67849 CEU87Z 136245089 IC50 = 580 nM T67849 CI6HG4 136249373 IC50 = 449 nM T67849 CL4MO3 136249382 IC50 = 278 nM T67849 C04LZP 136254186 IC50 = 29730 nM T67849 C8PT7R 136254187 IC50 > 100000 nM T67849 CCJV79 136254188 IC50 > 100000 nM T67849 C5QE8W 136254189 IC50 = 18970 nM T67849 C0GZV9 136254283 IC50 = 2870 nM T67849 CMWA86 136264282 IC50 = 36 nM T67849 CSD78N 136264452 IC50 = 1530 nM T67849 C1HI5T 136264454 IC50 = 21 nM T67849 CV3UE9 137333450 EC50 = 4.3 nM T67849 CH8WU5 137348751 IC50 = 0.7943 nM T67849 CH24ZD 137631369 IC50 = 2.4 nM T67849 CP34TI 137631388 IC50 = 7.4 nM T67849 CF0PQ2 137632018 IC50 = 1.585 nM T67849 C3XH0L 137632431 IC50 > 300 nM T67849 CF4JC7 137632807 IC50 = 110 nM T67849 CIX4S7 137633081 IC50 = 0.7943 nM T67849 CPG41O 137633365 IC50 = 120 nM T67849 C3ST1Q 137633684 IC50 = 1.259 nM T67849 CQ48RD 137633874 IC50 < 0.3 nM T67849 CA4MB6 137633919 IC50 = 10.7 nM T67849 CZ8Q6V 137634548 IC50 = 7200 nM T67849 CGO01Z 137634959 IC50 = 141 nM T67849 C9GXM1 137635017 IC50 = 1 nM T67849 C06BDR 137635072 IC50 = 11 nM T67849 CY86AJ 137635564 IC50 = 19.95 nM T67849 C5GHK7 137635800 IC50 = 16.8 nM T67849 CYK6C4 137635941 IC50 = 1 nM T67849 CMN6T7 137636115 IC50 = 6.73 nM T67849 CZ74XF 137636132 IC50 = 1.259 nM T67849 CPJ43Y 137636841 IC50 = 9.8 nM T67849 C1PVW6 137637361 IC50 > 300 nM T67849 CXPI97 137637422 IC50 = 6.31 nM T67849 CP2J4D 137638455 IC50 = 97.7 nM T67849 C83VBZ 137639018 IC50 = 6.6 nM T67849 CMZV19 137639099 IC50 = 1 nM T67849 CJ3LX4 137639119 IC50 = 9.4 nM T67849 CS78JW 137639139 IC50 = 16 nM T67849 CM4HB3 137639229 IC50 = 4.3 nM T67849 C8A2SJ 137639272 IC50 > 300 nM T67849 C4U8LN 137639297 IC50 = 9.6 nM T67849 C1UZ4S 137639310 IC50 = 44 nM T67849 CBK6W4 137639515 IC50 = 10100 nM T67849 CY52QL 137639725 IC50 = 2700 nM T67849 C4TSZ8 137639858 IC50 = 3.981 nM T67849 CKI6W2 137640126 IC50 = 240 nM T67849 C9EN8L 137640131 IC50 = 4.2 nM T67849 C7HA4V 137640279 IC50 = 10 nM T67849 CA0QO6 137640453 IC50 = 3.82 nM T67849 C37IUP 137640698 IC50 = 2700 nM T67849 C67NLM 137640896 IC50 = 12.59 nM T67849 CPW4L0 137641184 IC50 = 440 nM T67849 C2M1DL 137641375 IC50 = 3070 nM T67849 CQ8X0E 137641383 IC50 = 34 nM T67849 C0I6RQ 137641405 IC50 = 10 nM T67849 C8N1XG 137641715 IC50 = 135 nM T67849 CN3F5A 137641753 IC50 = 1.995 nM T67849 CLA7J8 137642251 IC50 = 12.2 nM T67849 C5X3TH 137642662 IC50 = 29 nM T67849 C8M9TX 137642801 IC50 = 29 nM T67849 CL4Q9G 137643238 IC50 = 2.512 nM T67849 CKU69P 137643285 IC50 = 50.12 nM T67849 CP3JK1 137643598 IC50 = 19.95 nM T67849 CE79MN 137643690 IC50 = 112 nM T67849 CV97OC 137644428 IC50 = 100 nM T67849 CAPQ93 137644458 IC50 = 20 nM T67849 CQSG70 137644855 IC50 = 107 nM T67849 C80WHF 137645205 IC50 = 620 nM T67849 CMYG31 137645705 IC50 = 43 nM T67849 CX8R1L 137645813 IC50 = 188 nM T67849 CID85J 137646014 IC50 = 70 nM T67849 C6SW7U 137646075 IC50 = 1.995 nM T67849 C5ERV3 137646413 IC50 = 27 nM T67849 CZC27Y 137646667 IC50 = 2.512 nM T67849 C3BM5S 137646790 IC50 = 1.4 nM T67849 CA4V8H 137646998 IC50 = 2.512 nM T67849 C9U0CF 137647045 IC50 = 5800 nM T67849 C5HIM9 137647114 IC50 = 2.512 nM T67849 CPMG65 137647250 IC50 = 0.87 nM T67849 C9K7OS 137647525 IC50 = 150 nM T67849 C3TXN9 137647591 IC50 = 13.8 nM T67849 CPX42N 137647765 IC50 = 15 nM T67849 C1FV9C 137647875 IC50 = 0.8 nM T67849 CI3UE7 137647995 IC50 = 41.5 nM T67849 CS39XP 137648085 IC50 = 1.585 nM T67849 C4Z0NQ 137648826 IC50 = 0.7943 nM T67849 CE54DO 137648917 IC50 = 5.012 nM T67849 CSML14 137649696 IC50 = 3 nM T67849 C9FAK1 137650131 IC50 = 0.3 nM T67849 C1R2BI 137650375 IC50 > 300 nM T67849 CUC02Z 137650404 IC50 = 5680 nM T67849 CHT1R8 137650579 IC50 = 2.512 nM T67849 CM8HZ3 137650719 IC50 = 1 nM T67849 CQ3KH9 137650741 IC50 = 4000 nM T67849 C5WR6T 137651215 IC50 = 0.9 nM T67849 CVEL76 137651324 IC50 = 2800 nM T67849 CS2RU9 137652004 IC50 = 170 nM T67849 C7PL6S 137652682 IC50 = 1.3 nM T67849 C9QA0W 137652944 IC50 = 12.59 nM T67849 C38FXZ 137653443 IC50 < 0.2 nM T67849 C1K6TD 137653515 IC50 = 11.8 nM T67849 CN78RE 137653565 IC50 = 0.7943 nM T67849 CTKQ38 137653713 IC50 = 39.81 nM T67849 CI26PN 137653800 IC50 = 9200 nM T67849 C13JPX 137654370 IC50 < 0.3 nM T67849 C9O7ZD 137654904 IC50 > 300 nM T67849 CD19ZS 137654937 IC50 = 4.9 nM T67849 C4N5LS 137655123 IC50 = 7.943 nM T67849 C29HVQ 137655302 IC50 = 4.5 nM T67849 CJNL46 137655684 IC50 = 1.4 nM T67849 CP4S1L 137655824 IC50 = 11.5 nM T67849 CHV26G 137655828 IC50 = 1.1 nM T67849 CC5NK4 137655965 IC50 = 2.512 nM T67849 C5T9JU 137656472 IC50 = 20 nM T67849 CLC7N4 137656507 IC50 = 1.585 nM T67849 CE9H8D 137657006 IC50 = 3.981 nM T67849 C1YN2Q 137657270 IC50 = 78.1 nM T67849 C1K4TB 137657388 IC50 = 14700 nM T67849 C2JX1W 137657572 IC50 = 3.162 nM T67849 C2D0TG 137657839 IC50 = 19.6 nM T67849 C41OPW 137658031 IC50 = 19.95 nM T67849 C6IR2E 137658119 IC50 = 2700 nM T67849 CU15TO 137658167 IC50 = 107 nM T67849 CCX72Y 137658365 IC50 = 60.2 nM T67849 C6BF8E 137658458 IC50 = 23 nM T67849 CI10RD 137658475 IC50 = 30 nM T67849 C90PIR 137658553 IC50 = 2900 nM T67849 CSB1U0 137658705 IC50 = 0.4 nM T67849 C03QAR 137659338 IC50 = 96.8 nM T67849 C5T8OX 137659620 IC50 > 300 nM T67849 C3CF4O 137659746 IC50 = 6.31 nM T67849 C49BSM 137659860 IC50 = 67.1 nM T67849 C1F6QN 137660818 IC50 = 1.259 nM T67849 C34WTV 137660874 IC50 = 5 nM T67849 CP5K4E 137660883 IC50 = 7.1 nM T67849 C1OLQ3 137660961 IC50 = 3.162 nM T67849 CM6FS2 137661095 IC50 = 1.585 nM T67849 C8R3JK 137661301 IC50 = 0.631 nM T67849 C6KR2A 137661344 IC50 = 80.2 nM T67849 C9HPG8 137661516 IC50 = 120 nM T67849 CKDZ26 138504497 IC50 = 800 nM T67849 C2T8OY 138857923 IC50 = 10 nM T67849 CPQ87J 139410792 IC50 < 20 nM T67849 C7ZAQ1 141406387 IC50 = 38160 nM T67849 C7NUI8 141406388 IC50 = 67810 nM T67849 CQYI18 141406390 IC50 = 11160 nM T67849 CUA1D0 141406392 IC50 = 56190 nM T67849 CP0R6Y 141406393 IC50 = 3910 nM T67849 C1EVQ0 141406394 IC50 = 23680 nM T67849 C2QP0F 141406396 IC50 = 44740 nM T67849 CY2M0B 141406399 IC50 = 8140 nM T67849 CC3OU2 141406400 IC50 = 47920 nM T67849 CKV13Y 141406404 IC50 = 28610 nM T67849 C3Q1VL 141419885 IC50 = 2.7 nM T67849 C3FPW6 141419887 IC50 = 7.8 nM T67849 C3EJX8 141419888 IC50 = 3.1 nM T67849 CKX4P3 141446054 IC50 = 7943.28 nM T67849 CV54CS 141471198 IC50 = 4.2 nM T67849 C25HYI 141471200 IC50 = 2.7 nM T67849 CZS03J 141509623 IC50 = 275 nM T67849 CFD94N 141754136 IC50 = 0.7 nM T67849 CX0E9B 142505968 IC50 = 68 nM T67849 C9G5ZW 142505990 IC50 = 5 nM T67849 CBJC50 142505992 IC50 = 49 nM T67849 CJ5GT3 142506013 IC50 = 0.7 nM T67849 C7N8LV 142506025 IC50 = 46 nM T67849 CKBF56 142506033 IC50 < 5 nM T67849 CQ34YR 142506035 IC50 = 81 nM T67849 CU03GW 142506036 IC50 = 4 nM T67849 C74MXW 142506065 IC50 = 0.7 nM T67849 C1PNM8 142506077 IC50 = 663 nM T67849 CX6BQ7 142506102 IC50 = 0.2 nM T67849 CY3BM0 142506119 IC50 = 96 nM T67849 CFJ6X3 142506136 IC50 = 133 nM T67849 CC6MD0 142506155 IC50 = 5 nM T67849 C05QOM 142506157 IC50 = 41 nM T67849 CLND62 142506170 IC50 = 520 nM T67849 CGNQ74 142506189 IC50 = 47 nM T67849 CT3U9R 142506192 IC50 = 0.2 nM T67849 CP71ZJ 142506208 IC50 = 189 nM T67849 C1T3IQ 142506210 IC50 = 0.2 nM T67849 CEGV67 142506220 IC50 = 0.6 nM T67849 CP5HF8 142506225 IC50 = 49 nM T67849 C1U3CA 142506238 IC50 = 32 nM T67849 C7QMG9 145108300 IC50 = 6.8 nM T67849 CGF4I3 145946093 IC50 = 5.012 nM T67849 CJ70MV 145946114 IC50 = 1 nM T67849 CI40JE 145951013 IC50 = 25.6 nM T67849 C6YT8E 145951131 IC50 = 5390 nM T67849 CFW62M 145951569 IC50 = 5.3 nM T67849 CHA84K 145951830 IC50 = 420.4 nM T67849 CT4I9A 145952160 IC50 = 53.9 nM T67849 C91GVH 145952598 IC50 = 1 nM T67849 C1W0GJ 145952796 IC50 = 19952.62 nM T67849 CY18SN 145953214 Ki = 20 nM T67849 CVMF13 145953272 IC50 = 2134 nM T67849 CYL5T1 145953372 IC50 <= 10000 nM T67849 CP14AV 145953653 IC50 = 751 nM T67849 CY8D5Q 145953886 IC50 = 10 nM T67849 C3ZUW8 145954195 IC50 = 156.5 nM T67849 C1NJB7 145955070 IC50 = 3 nM T67849 CRHE01 145955133 IC50 <= 10000 nM T67849 C7MP9Z 145955279 IC50 = 1.4 nM T67849 C7K8VT 145955565 IC50 = 6.2 nM T67849 CPU4X2 145955670 IC50 = 100.4 nM T67849 C3ST5Y 145955693 IC50 = 2 nM T67849 C1VH5X 145955836 IC50 = 20.5 nM T67849 CGHE02 145956080 Ki = 12 nM T67849 C7K2YF 145956631 IC50 <= 10000 nM T67849 CQW74M 145956683 IC50 = 3.3 nM T67849 CJ1F6A 145956725 IC50 = 135.2 nM T67849 C12IFO 145956886 IC50 = 8.6 nM T67849 C9O2PL 145958063 IC50 = 3.2 nM T67849 CQH01X 145958257 IC50 <= 10000 nM T67849 C3DGU7 145958571 IC50 = 1.3 nM T67849 C9NS6T 145958690 IC50 = 11.5 nM T67849 C7ZO9V 145959196 IC50 = 109.4 nM T67849 CSC81H 145959429 IC50 = 2.1 nM T67849 C0S1YM 145959980 IC50 = 21 nM T67849 CT3I2R 145960112 IC50 = 100 nM T67849 C8MJ9X 145960272 IC50 = 15 nM T67849 CF36RA 145961004 IC50 = 2 nM T67849 CHF56O 145961403 IC50 = 374 nM T67849 C2GT9Y 145961404 IC50 = 65 nM T67849 CAI0D6 145963117 IC50 = 87.8 nM T67849 CG6FW9 145967821 IC50 = 4.4 nM T67849 C9NH1Z 145967866 IC50 = 18.7 nM T67849 CCPB17 145967913 IC50 = 2.9 nM T67849 CB43FK 145968534 IC50 = 3 nM T67849 CGL03I 145969468 IC50 = 4.6 nM T67849 C2MST5 145969505 IC50 = 13.5 nM T67849 C97IKW 145969580 IC50 = 4.5 nM T67849 CK82QG 145969816 IC50 = 4364 nM T67849 C71YAK 145970017 IC50 = 10000 nM T67849 CKVI18 145970638 IC50 = 5.5 nM T67849 CTQ50N 145970860 IC50 = 5.5 nM T67849 CZ98FH 145971490 IC50 = 291.5 nM T67849 CTB97Z 145971948 IC50 = 11.5 nM T67849 CGQJ04 145972017 IC50 = 375.9 nM T67849 CA7X9N 145973949 IC50 = 307 nM T67849 CZ9G6E 145974533 IC50 = 12.3 nM T67849 C3LR4O 145976442 IC50 = 8672 nM T67849 CPZS56 145982349 EC50 = 19100 nM T67849 C3UWH8 145982505 IC50 = 84 nM T67849 C9UB4R 145982673 IC50 = 81 nM T67849 COI5P8 145982999 IC50 = 106 nM T67849 CH90CT 145983168 IC50 = 425.2 nM T67849 C1GLK2 145983578 IC50 = 86 nM T67849 CJU02I 145983624 IC50 = 8.4 nM T67849 CVS2U0 145983808 IC50 = 8.6 nM T67849 C6QL4V 145983880 IC50 = 16 nM T67849 CL6HZ9 145983897 IC50 = 227 nM T67849 CL0ZO7 145984847 IC50 = 26 nM T67849 CBTH68 145985019 IC50 = 41 nM T67849 C1HO7R 145986167 IC50 = 31 nM T67849 CP0IX3 145986185 IC50 = 416 nM T67849 CF8MR5 145986347 IC50 = 5000 nM T67849 C06ELG 145987952 IC50 = 3.4 nM T67849 CF82DR 145988183 IC50 = 8.1 nM T67849 CN0DH1 145989043 IC50 = 5.2 nM T67849 C6XMQ8 145989163 EC50 = 15670 nM T67849 CP8TH4 145989722 IC50 = 17 nM T67849 C8X2IT 145996536 IC50 = 1700 nM T67849 C6RPG0 146014481 IC50 = 7.413 nM T67849 C59KOM 146585662 IC50 = 7 nM T67849 CFQO97 146585699 IC50 = 60 nM T67849 C0GMR1 146585718 IC50 = 26 nM T67849 CI85VS 146731761 IC50 = 120 nM T67849 C4MC0S 149169124 IC50 = 4620 nM T67849 CVW62P 149242889 IC50 = 23680 nM T67849 CN87RZ 149370890 IC50 = 1420 nM T67849 CK4FJ1 149556361 IC50 = 7510 nM T67849 C8UQL4 153940691 IC50 = 750 nM T67849 CMZ68Q 153940692 IC50 = 420 nM T67849 C5X7JK 154734328 IC50 = 10 nM T67849 C69VNW 155510695 IC50 = 1584.89 nM T67849 C8Q9UG 155510876 IC50 = 390 nM T67849 CDT8F2 155510913 IC50 = 251.19 nM T67849 CQP9K0 155510991 IC50 = 970 nM T67849 CT6WX1 155511199 IC50 = 32 nM T67849 C9ZL7Y 155511258 IC50 = 11 nM T67849 CH12LB 155511310 IC50 = 374 nM T67849 C1OR2T 155511706 IC50 = 1000 nM T67849 C6PZ9F 155511758 IC50 = 540 nM T67849 C6WIC9 155511977 IC50 = 316.23 nM T67849 CPH8N1 155512095 IC50 = 3.162 nM T67849 CVX7Y0 155512208 IC50 = 33 nM T67849 CZJ9D6 155512258 IC50 = 24 nM T67849 CG9I4X 155512515 IC50 = 230 nM T67849 CR1Z8A 155512529 IC50 = 38 nM T67849 CD36LK 155512654 IC50 = 42 nM T67849 CQZY50 155512775 IC50 = 6.31 nM T67849 C5V2GO 155512947 IC50 = 398.11 nM T67849 C5GWL0 155513019 IC50 = 0.99 nM T67849 C1DIT4 155513047 IC50 = 50.12 nM T67849 C8PG6Z 155513084 IC50 = 158.49 nM T67849 C5M6NS 155513226 IC50 = 9.5 nM T67849 CZG6K5 155513391 IC50 = 60 nM T67849 C45SYX 155513615 IC50 = 2.2 nM T67849 C4UZI2 155514046 IC50 = 31622.78 nM T67849 C96VIE 155514302 IC50 = 11 nM T67849 CB81DS 155514349 IC50 = 6.2 nM T67849 C34VCY 155514382 IC50 = 8.4 nM T67849 CQ1X6F 155514587 IC50 = 42 nM T67849 CBH57O 155514764 IC50 = 125.89 nM T67849 C5C9EG 155515047 IC50 = 79.43 nM T67849 CEFS61 155515135 IC50 = 4720 nM T67849 CR1XO3 155515353 IC50 = 1258.93 nM T67849 C0AXF7 155515394 IC50 = 199.53 nM T67849 CXTC52 155515425 IC50 = 12589.25 nM T67849 CN1T7S 155515661 IC50 = 163 nM T67849 C7Q3FR 155515734 IC50 = 79.43 nM T67849 CL45GQ 155516260 IC50 = 1000 nM T67849 C5IR0K 155516391 IC50 = 2.4 nM T67849 C30ZFN 155516445 IC50 = 316.23 nM T67849 CJDG04 155516604 IC50 = 15.85 nM T67849 CRPB20 155516993 IC50 = 689 nM T67849 C42JXQ 155517064 IC50 = 199.53 nM T67849 CYO19V 155517071 IC50 = 158.49 nM T67849 CVY7O4 155517153 IC50 = 1.8 nM T67849 CYWX76 155517213 IC50 = 50.12 nM T67849 COE6G3 155517381 IC50 = 38 nM T67849 C0D3NR 155517424 IC50 = 25118.86 nM T67849 CT53XD 155517442 IC50 = 1584.89 nM T67849 C4G8YN 155517534 IC50 = 57 nM T67849 CS2JT9 155518175 IC50 = 1995.26 nM T67849 CW9GU4 155518188 IC50 = 1.7 nM T67849 CW7OM6 155518918 IC50 = 44 nM T67849 CC51GM 155519635 IC50 = 79.43 nM T67849 CMB6L0 155519660 IC50 = 343 nM T67849 CHFJ25 155519726 IC50 = 3.162 nM T67849 CZ78HW 155519830 IC50 = 79.43 nM T67849 CQEK39 155520373 IC50 = 6.8 nM T67849 C62TIK 155520386 IC50 = 29 nM T67849 C3D7FJ 155520444 IC50 = 3.162 nM T67849 C46YUA 155521057 IC50 = 87 nM T67849 C5D6YX 155521099 IC50 = 8100 nM T67849 C9N0YC 155521102 IC50 = 1.9 nM T67849 CEA3M1 155521494 IC50 = 25.12 nM T67849 CQD23C 155521715 IC50 = 2 nM T67849 CYI0T6 155521865 IC50 = 94 nM T67849 CBSR95 155522042 IC50 = 9490 nM T67849 CZO7Q8 155522149 IC50 = 44 nM T67849 CY0HL3 155522306 IC50 = 37 nM T67849 CCGW06 155523124 IC50 = 125.89 nM T67849 CNB70P 155523246 IC50 = 398.11 nM T67849 C4TLQ7 155523447 IC50 = 7 nM T67849 CO4S8X 155523501 IC50 > 10000 nM T67849 CZG27I 155523570 IC50 = 421 nM T67849 C37RVF 155523599 IC50 = 64 nM T67849 C4H2AB 155524238 IC50 = 12.59 nM T67849 CP18VT 155524467 IC50 = 12.59 nM T67849 C2PJ0X 155524583 IC50 = 89 nM T67849 C9VN1E 155524769 IC50 = 530 nM T67849 CUP7L2 155524901 IC50 = 100 nM T67849 C2BL5I 155525312 IC50 = 5.012 nM T67849 CE2OM4 155525333 IC50 = 3981.07 nM T67849 C10RZQ 155525477 IC50 = 19.95 nM T67849 CF76OV 155525717 IC50 = 3.9 nM T67849 CV21MY 155525971 IC50 = 39 nM T67849 C0UA4D 155525996 IC50 = 39.81 nM T67849 C0AR4W 155526097 IC50 = 5011.87 nM T67849 CD53VX 155526104 IC50 = 6.8 nM T67849 CNHS85 155526193 IC50 = 7943.28 nM T67849 C3EAR8 155526323 IC50 = 31.62 nM T67849 CFSJ40 155526749 IC50 = 0.93 nM T67849 CFHZ79 155527103 IC50 = 45 nM T67849 CK73QV 155527272 IC50 = 4.7 nM T67849 COU62P 155527495 IC50 = 31 nM T67849 C82NUW 155527501 IC50 = 38 nM T67849 CK07GS 155527559 IC50 = 38 nM T67849 CX12MK 155527651 IC50 = 4 nM T67849 CD89EL 155528247 IC50 = 3 nM T67849 CB9IO8 155528449 IC50 = 20 nM T67849 C8Z3TK 155528581 IC50 = 63.1 nM T67849 C0B2NV 155528644 IC50 = 3.2 nM T67849 COY5G1 155528831 IC50 = 58 nM T67849 CF1MS3 155528972 IC50 = 28.3 nM T67849 C3VAI9 155528997 IC50 = 251.19 nM T67849 C2FE1S 155529479 IC50 = 7.943 nM T67849 CB90AR 155529643 IC50 = 125.89 nM T67849 CFV1S0 155529706 IC50 = 40 nM T67849 C3XLY2 155529766 IC50 = 153 nM T67849 C14QOF 155530163 IC50 = 25.12 nM T67849 C4I5UP 155530224 IC50 = 158.49 nM T67849 CZL26X 155530501 IC50 = 18 nM T67849 CW24QE 155531054 IC50 = 576 nM T67849 CX6N3Y 155531155 IC50 = 79.43 nM T67849 C9AXO7 155531257 IC50 = 79.43 nM T67849 CGAI60 155531409 IC50 = 3.981 nM T67849 CDI4V8 155531526 IC50 = 34 nM T67849 CE6QP1 155532037 IC50 = 10 nM T67849 CJH9U4 155532237 IC50 = 1258.93 nM T67849 C6W0JX 155532471 IC50 = 501.19 nM T67849 CIM18N 155532540 IC50 = 28 nM T67849 CKMD29 155532546 IC50 = 125.89 nM T67849 CNMC95 155532794 IC50 = 11.1 nM T67849 C3XFB8 155532820 IC50 = 12.59 nM T67849 C0GR1J 155533050 IC50 = 0.7 nM T67849 CQS8P1 155533070 IC50 = 125.89 nM T67849 C0SZR9 155533335 IC50 = 150 nM T67849 CAT9V1 155533370 IC50 = 3 nM T67849 C67ERP 155533384 IC50 = 100 nM T67849 CL8OM7 155533564 IC50 = 4 nM T67849 CBM24U 155533579 IC50 = 125.89 nM T67849 CR5H8B 155533591 IC50 = 79.43 nM T67849 CA7T0Y 155533911 IC50 > 10000 nM T67849 C8XQ4W 155534168 IC50 = 0.2 nM T67849 CN1ST4 155534269 IC50 = 39.81 nM T67849 CDQY81 155534313 IC50 = 4 nM T67849 CBEG39 155534594 IC50 = 199.53 nM T67849 C3MT9C 155534643 IC50 = 150 nM T67849 C59SQY 155534735 IC50 = 27 nM T67849 CCXP81 155535236 IC50 = 180 nM T67849 CG1JR7 155535513 IC50 = 501.19 nM T67849 CN6KJ5 155535520 IC50 = 12.59 nM T67849 C8N6MT 155535532 IC50 = 10000 nM T67849 C5F2TY 155535537 IC50 = 19.95 nM T67849 CKB2U4 155535691 IC50 = 39.81 nM T67849 CY7X3M 155535740 IC50 = 12.59 nM T67849 CUWE49 155535963 IC50 = 630.96 nM T67849 C70UDF 155536179 IC50 = 125.89 nM T67849 CEJ6L1 155536226 IC50 = 3.7 nM T67849 CNB24M 155536473 IC50 = 25.12 nM T67849 CI6L8Q 155536677 IC50 = 26 nM T67849 CDF3T9 155536730 IC50 = 22 nM T67849 C2CG1A 155537016 IC50 = 251.19 nM T67849 CSO87C 155537103 IC50 = 12 nM T67849 CS24EV 155537776 IC50 = 110 nM T67849 C34SNT 155537955 IC50 = 58 nM T67849 C8AJ6C 155538256 IC50 = 1.3 nM T67849 CQ1E6H 155538266 IC50 = 15.85 nM T67849 CZ19AN 155538609 IC50 = 171 nM T67849 CHR8M1 155538990 IC50 = 9760 nM T67849 CZ9B1L 155539017 IC50 = 2.8 nM T67849 CC1BG2 155539321 IC50 = 25 nM T67849 CF20PS 155539394 IC50 = 100 nM T67849 CUC3F8 155539997 IC50 = 3.2 nM T67849 CL8NI2 155540037 IC50 = 23 nM T67849 C8LKW4 155540264 IC50 = 25.12 nM T67849 CKX3G2 155540908 IC50 = 7.2 nM T67849 C6I5DK 155541290 IC50 = 501.19 nM T67849 CI8XL2 155541479 IC50 = 9.6 nM T67849 CECX47 155541544 IC50 = 1.585 nM T67849 C7A3SN 155541583 IC50 = 49 nM T67849 C2D4ZP 155541609 IC50 = 7943.28 nM T67849 C4FC0V 155541900 IC50 = 251.19 nM T67849 C57MVO 155542051 IC50 = 5011.87 nM T67849 CASE16 155542363 IC50 = 794.33 nM T67849 C8AXF9 155542633 IC50 = 398.11 nM T67849 C8OC2P 155542800 IC50 = 320 nM T67849 C42BIZ 155542813 IC50 = 1000 nM T67849 CTDQ52 155542836 IC50 = 398.11 nM T67849 CVNR95 155542898 IC50 = 5 nM T67849 C1SY0G 155543154 IC50 = 4.8 nM T67849 C1JRK8 155543277 IC50 = 25118.86 nM T67849 C7IWJ2 155543389 IC50 = 5.012 nM T67849 C1UNH0 155543517 IC50 = 1258.93 nM T67849 CZY0N4 155543588 IC50 = 0.7 nM T67849 C48KXS 155543644 IC50 = 34 nM T67849 CJB8C9 155543659 IC50 = 42 nM T67849 C3CN0A 155543674 IC50 = 7.943 nM T67849 C5MYJ2 155543736 IC50 = 7943.28 nM T67849 CVI3E5 155543933 IC50 = 0.43 nM T67849 C8OSM3 155544223 IC50 = 635 nM T67849 CX1C8I 155544561 IC50 = 8.5 nM T67849 COGF23 155544916 IC50 = 25118.86 nM T67849 C48RPZ 155544941 IC50 = 1000 nM T67849 C98FXC 155544955 IC50 = 50 nM T67849 CW3K4F 155545182 IC50 = 3162.28 nM T67849 C4TYN3 155545535 IC50 = 25118.86 nM T67849 CV8G5R 155545946 IC50 = 27 nM T67849 CTSW53 155546042 IC50 = 9.2 nM T67849 C1HKU0 155546330 IC50 = 33 nM T67849 CQ6J7U 155546361 IC50 = 990 nM T67849 CE1A0D 155546906 IC50 = 9.4 nM T67849 C8SQA2 155546999 IC50 = 6.31 nM T67849 C8D4ZH 155547166 IC50 = 316.23 nM T67849 CMY3J7 155547466 IC50 = 231 nM T67849 C2BS7T 155547557 IC50 = 1270 nM T67849 C31GSV 155547741 IC50 = 47 nM T67849 CH1F9K 155547869 IC50 = 5.9 nM T67849 CJAB13 155548110 IC50 = 18.4 nM T67849 CI6KO7 155548518 IC50 = 316.23 nM T67849 CL4F8P 155549003 IC50 = 6.31 nM T67849 CM6S8K 155549098 IC50 = 39.81 nM T67849 CON58B 155549407 IC50 = 27 nM T67849 CFMH09 155549542 IC50 = 179 nM T67849 C4PEJ5 155549895 IC50 = 9310 nM T67849 CFP94J 155550309 IC50 = 199.53 nM T67849 CCX5E2 155550788 IC50 = 180 nM T67849 CZS9Q8 155551405 IC50 = 0.7943 nM T67849 C3QZE7 155551609 IC50 = 20 nM T67849 CFO52S 155551740 IC50 = 252 nM T67849 C5HR2W 155551907 IC50 = 15848.93 nM T67849 CK1JR7 155551961 IC50 = 7.4 nM T67849 CK53PC 155552028 IC50 = 91 nM T67849 CI3Y5U 155552035 IC50 = 22 nM T67849 CUD43T 155552139 IC50 = 14.3 nM T67849 CWJ72T 155552555 IC50 = 220 nM T67849 CXN3Y8 155553327 IC50 = 25.12 nM T67849 CL04BD 155554125 IC50 = 37 nM T67849 CX9C6O 155554180 IC50 = 19.95 nM T67849 CP7L5X 155554538 IC50 = 14 nM T67849 CVH0M1 155554616 IC50 = 4.9 nM T67849 CC13QL 155555170 IC50 = 263 nM T67849 CZX06J 155555458 IC50 = 50.12 nM T67849 C2OGW1 155555483 IC50 = 29 nM T67849 C3UP9A 155555623 IC50 = 3981.07 nM T67849 C3KXR2 155555660 IC50 = 3 nM T67849 C19WIO 155555836 IC50 = 498 nM T67849 CRO5Z3 155556073 IC50 = 7 nM T67849 CH2P4T 155556124 IC50 = 158489.32 nM T67849 CCU8M1 155556480 IC50 = 501.19 nM T67849 CIU29Z 155556576 IC50 = 11 nM T67849 CM3LI6 155556593 IC50 = 143 nM T67849 CZ8CX1 155556887 IC50 = 39.81 nM T67849 CG2FS6 155557123 IC50 = 50.12 nM T67849 CFS63H 155557182 IC50 = 2 nM T67849 CCL48D 155557746 IC50 = 120 nM T67849 C0FE4G 155557988 IC50 = 170 nM T67849 CR8J0E 155558167 IC50 = 79.43 nM T67849 CN96JH 155558197 IC50 = 1000 nM T67849 CSO4M3 155558261 IC50 = 501.19 nM T67849 C52TSP 155558262 IC50 = 144 nM T67849 CB4A1O 155558535 IC50 = 1258.93 nM T67849 C2VGC6 155558733 IC50 = 7.7 nM T67849 CZMI26 155558737 IC50 = 15848.93 nM T67849 CDS2U1 155558931 IC50 = 24 nM T67849 CLS9Y1 155559053 IC50 = 61 nM T67849 CS70ER 155559192 IC50 = 163 nM T67849 C9KX4D 155559215 IC50 = 920 nM T67849 CSF7G4 155559324 IC50 = 2.5 nM T67849 CAQ0X8 155559376 IC50 = 29.4 nM T67849 CMKY39 155559468 IC50 = 15848.93 nM T67849 CAWI85 155559815 IC50 = 8.9 nM T67849 CDI59L 155560058 IC50 = 5.012 nM T67849 CDJ1P2 155560222 IC50 = 3.2 nM T67849 CVG49I 155560688 IC50 = 5450 nM T67849 C5S7AL 155560766 IC50 = 79.43 nM T67849 C2OT6K 155560767 IC50 = 3162.28 nM T67849 CQ7PS9 155560780 IC50 = 7.943 nM T67849 CLO3B1 155561152 IC50 = 20 nM T67849 C8XS0L 155561165 IC50 = 39.81 nM T67849 C72CQG 155561233 IC50 = 15.85 nM T67849 C1INL7 155561328 IC50 = 19.95 nM T67849 C98FHW 155561366 IC50 = 27 nM T67849 CUGI82 155561991 IC50 = 42 nM T67849 C35VQO 155562231 IC50 = 405 nM T67849 CB1T2W 155562315 IC50 > 31622.78 nM T67849 CX6U2T 155562388 IC50 = 79.43 nM T67849 CN4B3D 155562639 IC50 = 25118.86 nM T67849 C5E9TP 155562641 IC50 > 39810.72 nM T67849 CCF4W2 155563986 IC50 = 158.49 nM T67849 CVZ80N 155564202 IC50 = 10 nM T67849 CYD52H 155564883 IC50 = 178 nM T67849 CHK4E8 155565269 IC50 = 63.1 nM T67849 C7PXA0 155565551 IC50 = 6.31 nM T67849 CY4N7O 155565715 IC50 = 3981.07 nM T67849 CVQ6Z4 155565763 IC50 = 100 nM T67849 CA1RX3 155565771 IC50 = 251.19 nM T67849 CQ3AU4 155565828 IC50 = 630.96 nM T67849 CMK4I3 155565845 IC50 = 63.1 nM T67849 C59VPW 155565958 IC50 = 12.59 nM T67849 CAP9F2 155566187 IC50 = 3 nM T67849 CY5SB4 155566208 IC50 = 63.1 nM T67849 CM7E2G 155566279 IC50 = 794.33 nM T67849 C3BNY5 155566309 IC50 = 316.23 nM T67849 C9HR5K 155566863 IC50 = 15848.93 nM T67849 CXE94L 155567270 IC50 = 43 nM T67849 C9KQW3 155567372 IC50 = 14 nM T67849 C98NZE 155567616 IC50 = 19952.62 nM T67849 C1HQ5J 155568324 IC50 = 6.3 nM T67849 CLA46O 155568356 IC50 = 1780 nM T67849 CH2RY0 155568388 IC50 = 150 nM T67849 C7SLR8 155568452 IC50 = 6.31 nM T67849 CT15RN 155568479 IC50 = 1584.89 nM T67849 CM5XO0 155568497 IC50 = 8330 nM T67849 C3VTU8 155568539 IC50 = 1470 nM T67849 CT0BK2 155568581 IC50 = 11.4 nM T67849 C14LVO 155569074 IC50 = 125.89 nM T67849 CFWP17 155569113 IC50 = 22 nM T67849 C1UD4S 155569289 IC50 = 19.95 nM T67849 CXBZ67 155569362 IC50 = 12589.25 nM T67849 CUH38L 155569363 IC50 = 6150 nM T67849 C4H0NE 155569598 IC50 = 100 nM T67849 D00HSJ 10275789 IC50 = 910 nM T67849 D00ZIK 9908783 Ki = 20 nM T67849 D01SSI 24937012 IC50 = 15 nM T67849 D03EHM 24905142 IC50 = 150 nM T67849 D03QQH 16760391 IC50 = 22000 nM T67849 D06DNH 9907093 IC50 = 851 nM T67849 D06HVH 54613583 IC50 = 4700 nM T67849 D06PWI 42623951 IC50 = 7943.28 nM T67849 D07PMP 44187953 IC50 = 14 nM T67849 D08KSQ 11637090 IC50 > 10000 nM T67849 D08NQM 5289247 IC50 = 300 nM T67849 D0H2CM 135565635 IC50 = 100 nM T67849 D0P5TI 58441401 IC50 = 3020 nM T67849 D0R0TW 11964036 IC50 < 0.1 nM T67849 D0S5YV 6852167 IC50 = 77 nM T67849 D0W8XH 9884685 IC50 = 3 nM T67849 D0X1RH 16051023 IC50 = 440 nM T67849 D0Y3OO 11327430 IC50 = 30 nM T51426 D01VMO 3401 IC50 = 13800 nM T51426 D01XBA 5035 IC50 = 11560 nM T51426 D03ZTE 10133 EC50 = 3400 nM T51426 D04VIS 5318517 IC50 = 9700 nM T51426 D06ABF 3957 IC50 = 3070 nM T51426 D06RGG 5819 IC50 = 7860 nM T51426 D08QIP 4887 EC50 = 15000 nM T51426 D09GOS 2812 IC50 = 3240 nM T51426 D0G3SH 31401 EC50 > 50000 nM T51426 D0G8BV 6450278 Ki > 5000 nM T51426 D0JO7Y 104741 IC50 = 790 nM T51426 D0M4WA 447715 EC50 = 10 nM T51426 D0OR2L 221493 EC50 = 45000 nM T51426 D0WN0U 3333 IC50 = 4960 nM T51426 D0X8XA 5318 IC50 = 6880 nM T51426 D01SYU 10026128 EC50 = 4 nM T51426 D02PQB 222528 EC50 = 45000 nM T51426 D04SLF 9903 EC50 = 6700 nM T51426 D05EUR 121418176 EC50 = 0.5 nM T51426 D00UQF 9893571 EC50 = 15 nM T51426 D09FOM 42601440 EC50 = 280 nM T51426 D0R8GK 50943003 EC50 = 4 nM T51426 D0TH6M 25204767 EC50 = 121 nM T51426 D0YZ8I 4273754 IC50 = 3220 nM T51426 D0Y2IH 122023 IC50 = 35200 nM T51426 CY6VB8 107794 IC50 = 7920 nM T51426 CY6G0E 126016 EC50 = 16200 nM T51426 C9DK4X 136695 EC50 = 530 nM T51426 CC81NZ 363417 IC50 = 9750 nM T51426 CEX6R9 447718 EC50 = 1300 nM T51426 C2BJ7P 583994 IC50 = 16400 nM T51426 CRZB53 669716 EC50 = 1400 nM T51426 CG5D1Q 803886 EC50 = 410 nM T51426 C5G6QA 808655 EC50 = 4000 nM T51426 CP6Q5B 808754 EC50 = 160 nM T51426 CP8U1D 808816 EC50 = 560 nM T51426 CE9F4J 808820 EC50 = 1270 nM T51426 CA95UQ 808823 EC50 = 130 nM T51426 CKE01Q 808825 EC50 = 170 nM T51426 C0LM6P 808829 EC50 = 540 nM T51426 C8BA1P 808833 EC50 = 20 nM T51426 CTY73N 808837 EC50 = 310 nM T51426 C7M2YC 808854 EC50 = 250 nM T51426 CNH98L 836804 IC50 > 100000 nM T51426 CGUN17 836806 IC50 = 10200 nM T51426 C5SIF2 836814 IC50 > 100000 nM T51426 CGCM38 836818 IC50 > 100000 nM T51426 CD50VK 836830 IC50 > 100000 nM T51426 CN4R2H 836832 IC50 > 100000 nM T51426 CN5M0I 836845 IC50 > 100000 nM T51426 CNO02J 858049 EC50 = 170 nM T51426 CNFT92 877112 EC50 = 350 nM T51426 CP7RZ2 989521 EC50 = 5150 nM T51426 C0D8CN 1088402 EC50 = 5990 nM T51426 CGWD09 3205789 EC50 = 910 nM T51426 CM68NH 3205794 EC50 = 480 nM T51426 C98IRC 3311258 EC50 = 370 nM T51426 CBR07T 3973060 EC50 = 500 nM T51426 C62FMD 4230997 IC50 = 47 nM T51426 C1SD4X 4335872 EC50 = 24 nM T51426 CC2RL5 4799393 IC50 = 3770 nM T51426 C5BKQ7 5111487 IC50 = 76 nM T51426 CC8T0K 5152913 EC50 = 120 nM T51426 CM73PF 5220350 EC50 = 150 nM T51426 C09QOX 5284060 EC50 = 6000 nM T51426 C4EV1S 5284061 EC50 > 31600 nM T51426 CNA12W 5708333 IC50 = 20000 nM T51426 CT5B6O 5885580 EC50 = 1160 nM T51426 C5O9WK 6161915 IC50 = 4290 nM T51426 C16ZSG 6439929 EC50 = 130 nM T51426 CXY21G 6460218 EC50 = 2900 nM T51426 CSG96A 6461297 IC50 = 27000 nM T51426 CAD3B4 6611349 IC50 = 810 nM T51426 C6T9AD 9448220 IC50 = 20000 nM T51426 CMIW83 9812710 IC50 = 260 nM T51426 C9F7MT 9847547 EC50 = 3260 nM T51426 C7BEU4 9910920 EC50 > 100000 nM T51426 C2SHJ5 9911971 EC50 = 19 nM T51426 CN3WX7 9983614 EC50 = 29680 nM T51426 C2O3FL 10000577 EC50 = 57 nM T51426 CXR3V2 10003531 EC50 = 72 nM T51426 CPOA71 10005757 EC50 = 72 nM T51426 CTDH25 10025364 EC50 = 12 nM T51426 C89XQB 10027247 EC50 = 51 nM T51426 CAP62L 10028914 EC50 = 69 nM T51426 CIX7D6 10050542 EC50 = 206 nM T51426 C4ASR3 10070121 EC50 = 32 nM T51426 C8XZ7P 10074158 EC50 = 6000 nM T51426 CJ14SF 10097386 EC50 = 64 nM T51426 C2S7CM 10117653 EC50 = 38 nM T51426 C0AC6X 10206024 EC50 = 36 nM T51426 CVWU14 10255620 EC50 = 66 nM T51426 CL72TC 10321416 EC50 = 77 nM T51426 C6D5LO 10343437 IC50 = 60400 nM T51426 CNF86C 10366850 EC50 = 70 nM T51426 CV7B2U 10386768 EC50 = 73 nM T51426 CKET62 10405361 IC50 = 3100 nM T51426 CRZ01P 10436479 EC50 = 77 nM T51426 CZ29PD 10477364 EC50 = 25 nM T51426 CZJ0F4 10479213 EC50 = 57 nM T51426 CI1G2S 10479586 EC50 > 100000 nM T51426 C2P4FZ 10506710 EC50 = 48 nM T51426 CGX0L9 10554022 EC50 = 47 nM T51426 CNZ48O 10572244 IC50 = 31600 nM T51426 CN5QH7 10578428 EC50 = 60 nM T51426 CY3BQ1 10603436 EC50 = 12 nM T51426 CEZ2B4 10612087 IC50 = 15100 nM T51426 C5TA6W 10625842 EC50 = 100 nM T51426 CG73DH 10649304 EC50 = 70 nM T51426 C1ZWP4 10715824 EC50 = 230 nM T51426 C9GMJ7 10744903 EC50 = 100 nM T51426 CRF9V2 10768688 EC50 = 37 nM T51426 CN94LQ 10840310 EC50 = 54 nM T51426 CYS74G 10862978 EC50 > 1000 nM T51426 C7LF4S 10863403 EC50 > 1000 nM T51426 C7PAN9 10863689 EC50 = 162.18 nM T51426 CQ9OW2 10863818 EC50 = 89 nM T51426 CHS76V 10863889 EC50 = 358 nM T51426 CP9ZK5 10864128 EC50 = 132 nM T51426 CU8I2C 10865031 EC50 = 1470 nM T51426 C1P6MD 10874384 EC50 = 96 nM T51426 CX49GE 10880703 EC50 > 1000 nM T51426 CL0G9X 10884439 EC50 = 163 nM T51426 CX74QO 10885046 EC50 = 198000 nM T51426 CQZG56 10885149 EC50 = 109 nM T51426 CPD79S 10895508 EC50 = 449 nM T51426 CWLA47 10895757 EC50 = 173 nM T51426 C5CK7U 10906872 EC50 = 108 nM T51426 CI0V2P 10907468 EC50 = 932 nM T51426 CYU0Z4 10918067 EC50 = 247 nM T51426 CM3S8H 10918117 EC50 = 256 nM T51426 C4FV5Q 10928377 EC50 = 377 nM T51426 CP9O6G 10929283 EC50 = 195 nM T51426 C3AX4K 10929645 EC50 = 1000 nM T51426 C15ZJA 10939815 EC50 = 77 nM T51426 C6AL9W 10939865 EC50 = 205 nM T51426 CF1O5U 10940474 EC50 = 416.87 nM T51426 C7A1CD 10951158 EC50 = 219 nM T51426 CO1E9F 10959425 EC50 = 10000 nM T51426 CFW15Y 10960421 IC50 = 75000 nM T51426 C5LE9H 10961580 EC50 = 1400 nM T51426 C73RAP 10961679 EC50 = 343 nM T51426 CM9I4X 10974102 EC50 > 1000 nM T51426 CW4UR6 10983879 EC50 = 236 nM T51426 CFW6U7 10984625 EC50 = 333 nM T51426 CC0XW4 10993939 EC50 = 97 nM T51426 CC17TD 10994116 EC50 > 1000 nM T51426 CC98JZ 10994566 EC50 > 1000 nM T51426 C6CR4P 10995572 EC50 > 1000 nM T51426 C53JGN 11005354 EC50 = 149 nM T51426 CB9V8P 11006123 EC50 > 1000 nM T51426 CG54EL 11006667 EC50 > 1000 nM T51426 C4NI7K 11012074 EC50 > 1000 nM T51426 CMZI02 11016010 EC50 > 1000 nM T51426 CD7Y9V 11016217 EC50 > 1000 nM T51426 CRT5C1 11016287 EC50 = 212 nM T51426 C9UC1O 11016318 EC50 = 309 nM T51426 CB1FT9 11016535 EC50 = 185 nM T51426 CPG87I 11016574 EC50 = 227 nM T51426 CCVO17 11026506 EC50 = 602.56 nM T51426 CKA98L 11026848 EC50 > 1000 nM T51426 C3UGS5 11027458 EC50 = 147 nM T51426 CNQ2G9 11037825 EC50 = 71 nM T51426 CG4LT7 11037848 EC50 = 1370 nM T51426 C8SRF7 11038288 EC50 = 243 nM T51426 C1MO8H 11049585 EC50 = 233 nM T51426 C9AJ4F 11049685 EC50 > 1000 nM T51426 CV2E8L 11049902 EC50 = 150 nM T51426 CPM86Q 11059371 EC50 = 1000 nM T51426 C14SZU 11059537 EC50 = 120 nM T51426 CQI75L 11069965 EC50 = 118 nM T51426 CZ4K3C 11070729 EC50 = 162 nM T51426 CJ2BK9 11070754 EC50 = 95 nM T51426 CT2BZ5 11071069 EC50 = 227 nM T51426 C1V3OW 11071316 EC50 = 165 nM T51426 C1FD9O 11072109 EC50 > 1000 nM T51426 CN8Y7T 11091466 EC50 = 310 nM T51426 CAY09B 11091792 EC50 = 228 nM T51426 C7O4LY 11092153 EC50 = 561 nM T51426 C91KZB 11100907 EC50 > 1000 nM T51426 CF0EL5 11101594 EC50 > 1000 nM T51426 C7M1QZ 11102779 EC50 = 431 nM T51426 C1V8FP 11102780 EC50 = 467 nM T51426 C8U5MB 11103071 EC50 = 431 nM T51426 CH5UI7 11103128 EC50 > 1000 nM T51426 C16UHD 11103317 EC50 = 1000 nM T51426 CH43EJ 11113376 EC50 = 128.82 nM T51426 CJI3A0 11114198 EC50 > 1000 nM T51426 C3TZY0 11123056 EC50 = 64.57 nM T51426 C0GZJ1 11123604 EC50 > 1000 nM T51426 CM5J6E 11134927 EC50 = 220 nM T51426 C1V9PQ 11135300 EC50 = 263.03 nM T51426 CQE57C 11145151 EC50 = 348 nM T51426 C23PZQ 11145640 EC50 = 208 nM T51426 C8GEB4 11146134 EC50 > 1000 nM T51426 CPJK71 11155112 EC50 = 1220 nM T51426 C9ND0W 11187621 EC50 = 210 nM T51426 CYS87Q 11292616 EC50 = 60 nM T51426 COLQ57 11731226 EC50 > 1000 nM T51426 CR3N9H 11733774 EC50 = 86 nM T51426 CE5IV9 11734521 EC50 = 1950 nM T51426 CRO02H 11750111 EC50 = 22 nM T51426 C9B6XF 11750447 EC50 = 29 nM T51426 CY1T9K 11751452 EC50 = 45 nM T51426 CI5C3B 11762020 EC50 = 1318.26 nM T51426 CHE2O5 11762919 EC50 = 267 nM T51426 CKFD53 11812810 EC50 = 226 nM T51426 CIVD16 11812930 EC50 = 94 nM T51426 CXO93Q 11826446 EC50 = 233 nM T51426 CUDK36 12369941 EC50 = 6170 nM T51426 CS3L4D 14036811 EC50 = 3570 nM T51426 CL6Z5O 14036813 EC50 = 2100 nM T51426 COV90A 14233056 EC50 = 15000 nM T51426 CWC43V 14820108 IC50 > 100000 nM T51426 CY2Z4L 15558616 EC50 = 10160 nM T51426 CJ9NC0 15558620 EC50 = 8800 nM T51426 C8HYN2 15604877 EC50 = 3400 nM T51426 CIH2Y5 16034640 EC50 = 460 nM T51426 CL8SW3 16049773 IC50 = 8100 nM T51426 C3BQ1I 16138920 IC50 = 500 nM T51426 CP2I4M 16178905 IC50 = 5000 nM T51426 CP7A5G 16392922 IC50 = 3300 nM T51426 CV63ZY 16579168 IC50 = 11800 nM T51426 C2HLZ9 16660329 IC50 = 1 nM T51426 CSXO69 16680454 EC50 = 200 nM T51426 C08HCW 17171885 EC50 = 320 nM T51426 C3T1KI 17171912 EC50 = 440 nM T51426 CY8HU9 17171920 EC50 = 1360 nM T51426 CJ0O5G 17341936 IC50 = 630 nM T51426 CWX3O9 17360242 EC50 = 370 nM T51426 C7B6AR 17556804 IC50 = 9400 nM T51426 C3E2KQ 17565898 IC50 = 1300 nM T51426 CG2KT4 17639891 EC50 = 160 nM T51426 CWA8J6 17755103 EC50 > 100000 nM T51426 C2LMW1 18565134 EC50 = 5900 nM T51426 C0QKH8 18565138 EC50 = 7600 nM T51426 CGS1R9 18565141 EC50 = 5300 nM T51426 C38JEL 20704150 EC50 = 9000 nM T51426 C35DEL 21121407 EC50 > 100000 nM T51426 CVR49B 21778740 IC50 = 24800 nM T51426 C8U7EC 21778741 IC50 = 64500 nM T51426 CU0I9S 24106478 IC50 = 970 nM T51426 CYS41V 24178657 IC50 > 100000 nM T51426 C8VYF7 24178772 IC50 = 24000 nM T51426 CWA5T3 24551913 EC50 = 14400 nM T51426 C53ISN 24739170 EC50 = 45 nM T51426 CKN7U1 24739171 EC50 = 420 nM T51426 C6LH0B 24739173 EC50 = 2300 nM T51426 CTE1N2 24748569 EC50 = 15 nM T51426 CMJ45V 24757189 EC50 = 3000 nM T51426 CFNW96 24757274 EC50 = 3100 nM T51426 CM5XR2 24757275 EC50 = 2100 nM T51426 C4DZA6 24757276 EC50 = 2500 nM T51426 CV4C1P 24757444 EC50 = 840 nM T51426 C85ELO 24771983 EC50 = 50 nM T51426 C3DH6Z 24776359 EC50 = 9000 nM T51426 CFP34W 24776360 EC50 = 35100 nM T51426 CM3AT1 24776361 EC50 = 1300 nM T51426 CIQ32L 24776362 IC50 = 15800 nM T51426 CG21UO 24776363 IC50 = 22200 nM T51426 C7N9XA 24776364 IC50 = 33900 nM T51426 C19PEN 24776365 EC50 = 1300 nM T51426 CS6JA4 24776366 IC50 = 4000 nM T51426 CJFQ78 24776367 IC50 = 3700 nM T51426 C3LN2R 24800409 IC50 = 70 nM T51426 C4UVQ7 25108827 EC50 = 20 nM T51426 CF5Z7J 25110740 EC50 = 1860 nM T51426 C6XF0P 25113666 EC50 = 32 nM T51426 C4C6YU 25117973 IC50 = 25300 nM T51426 C24YCZ 25118391 IC50 = 81100 nM T51426 CX9IR5 25121533 EC50 = 600 nM T51426 C5T7SP 25131364 EC50 = 88 nM T51426 C64VQS 25131696 EC50 = 51 nM T51426 C9F7EH 25131697 EC50 = 140 nM T51426 C3X7LV 25131698 EC50 = 490 nM T51426 CAFL43 25132042 EC50 = 670 nM T51426 CL43VE 25132043 EC50 = 21 nM T51426 CO7EX5 25132044 EC50 = 250 nM T51426 C0E8NR 25132408 EC50 = 550 nM T51426 C27TNZ 25132749 EC50 = 190 nM T51426 C0BH2Y 25132751 EC50 = 1200 nM T51426 C7W4CD 25165362 EC50 = 200 nM T51426 CP4T9S 25165363 EC50 = 150 nM T51426 CKJ21Q 25165364 EC50 = 410 nM T51426 CJC9M4 25165568 EC50 = 160 nM T51426 CF1NC8 25165571 EC50 = 160 nM T51426 C3A7RJ 25165769 EC50 = 440 nM T51426 C6A8XK 25166350 EC50 = 63 nM T51426 CCF9H7 25166548 EC50 = 380 nM T51426 CV8F9R 25166549 EC50 = 110 nM T51426 CZ5LX4 25166550 EC50 = 710 nM T51426 C71VLW 25166551 EC50 = 81 nM T51426 CRZ90W 25166552 EC50 = 1700 nM T51426 CH13FO 25166753 EC50 = 1400 nM T51426 CC4J0Q 25166754 EC50 = 160 nM T51426 CUW49M 25166755 EC50 = 670 nM T51426 C83XMC 25166756 EC50 = 1100 nM T51426 CD0CB8 25166970 EC50 = 1500 nM T51426 C79CVP 25167167 EC50 = 590 nM T51426 CTXL20 25167170 EC50 = 480 nM T51426 CDQ3N6 25167372 EC50 = 210 nM T51426 CCXL09 25167373 EC50 = 710 nM T51426 CG3BD7 25220917 EC50 = 900 nM T51426 CZ6TO8 25223264 EC50 = 500 nM T51426 CU5GV7 25223265 EC50 = 500 nM T51426 CYC03D 25223266 EC50 = 1100 nM T51426 C8G4WE 25223267 EC50 = 8 nM T51426 CS7E1J 25329558 EC50 = 4330 nM T51426 CTY7W5 25356628 IC50 = 8230 nM T51426 CT4P2K 25527221 EC50 = 2600 nM T51426 CFO6R7 25767966 IC50 = 680 nM T51426 CQ12AN 25767990 IC50 = 850 nM T51426 CW75TY 28759467 IC50 = 350 nM T51426 CO0J9C 36656496 IC50 = 6600 nM T51426 C2XZE6 42601492 EC50 = 2.5 nM T51426 CG6E4W 42611143 EC50 = 6.5 nM T51426 C80TIU 42611160 EC50 = 6.3 nM T51426 CK74NO 42611161 EC50 = 5 nM T51426 CP14GL 42611162 EC50 = 35 nM T51426 CU6W0Z 42611163 EC50 = 12 nM T51426 C86YDK 42611164 EC50 = 16 nM T51426 CTUZ74 42611165 EC50 = 8.5 nM T51426 CD1CN9 42628984 IC50 = 45 nM T51426 CJX95C 42738384 EC50 = 240 nM T51426 CJDV12 42738386 EC50 = 1900 nM T51426 C6D4WU 43911037 EC50 = 170 nM T51426 C0EIW1 44143573 EC50 = 10000 nM T51426 CDHU87 44143574 IC50 = 170 nM T51426 CN8K6B 44143575 EC50 = 52 nM T51426 CY0QM8 44143576 EC50 = 5000 nM T51426 CUK47P 44143577 IC50 = 1720 nM T51426 CXZD86 44143578 IC50 = 2750 nM T51426 CH67ZQ 44143579 EC50 = 4000 nM T51426 C5J2ZH 44143580 IC50 = 310 nM T51426 CCB2S7 44198477 IC50 = 1400 nM T51426 C5LI8K 44198480 IC50 = 60 nM T51426 C9S7FT 44198732 EC50 = 10600 nM T51426 C1KZL8 44399030 EC50 = 255000 nM T51426 C5A9KS 44399088 EC50 = 255000 nM T51426 CUG60W 44399191 EC50 = 222000 nM T51426 C7MLN5 44399399 EC50 = 680 nM T51426 C2K6ZW 44427760 EC50 > 100000 nM T51426 C8TYE6 44427761 EC50 = 11600 nM T51426 CI86EY 44427762 EC50 = 11800 nM T51426 C5K7DN 44427764 EC50 = 10500 nM T51426 CM02GU 44457471 EC50 > 100000 nM T51426 CQ21YX 44457491 EC50 = 10600 nM T51426 C2OI7T 44457500 EC50 > 31600 nM T51426 CK80JN 44457504 EC50 > 50000 nM T51426 CR5SI0 44476535 EC50 = 6 nM T51426 CW9T8Z 44573831 EC50 = 74 nM T51426 C7LK1S 44573832 EC50 = 720 nM T51426 C6LS4Z 44573833 EC50 = 480 nM T51426 CHOS17 44573862 EC50 = 620 nM T51426 CA83XI 44573942 EC50 = 900 nM T51426 CAEH73 44573943 EC50 = 1100 nM T51426 CK4WT5 44573944 EC50 = 1100 nM T51426 C27BAF 44573987 EC50 = 87 nM T51426 C18MCK 44573988 EC50 = 110 nM T51426 C72AMS 44573989 EC50 = 58 nM T51426 CZ8SH6 44574017 EC50 = 110 nM T51426 C9KHA0 44574018 EC50 = 930 nM T51426 CQ60ZF 44574019 EC50 = 960 nM T51426 C40WVF 44574040 EC50 = 930 nM T51426 CSWD46 44574041 EC50 = 2000 nM T51426 C34MYL 44574042 EC50 = 140 nM T51426 CK8H9V 44574071 EC50 = 240 nM T51426 C8MHU5 44574072 EC50 = 280 nM T51426 C9MPU7 44574073 EC50 = 190 nM T51426 C8JOM3 44574102 EC50 = 93 nM T51426 C4FRT2 44574173 EC50 = 230 nM T51426 CMC15E 44574174 EC50 = 93 nM T51426 CZ5GT2 44574199 EC50 = 1200 nM T51426 C6Q9GW 44574200 EC50 = 48 nM T51426 C6OF3T 44574201 EC50 = 600 nM T51426 CM9SI5 44574202 EC50 = 7800 nM T51426 CL0Y2T 44574231 EC50 = 1100 nM T51426 C2N4IC 44574232 EC50 = 78 nM T51426 C1AE6I 44574233 EC50 = 72 nM T51426 CTUI54 44574261 EC50 = 400 nM T51426 CVQ2W7 44574262 EC50 = 51 nM T51426 C84DKQ 44574263 EC50 = 28 nM T51426 CV9DO5 44574297 EC50 = 150 nM T51426 CP73NK 44574298 EC50 = 82 nM T51426 CYTB53 44574299 EC50 = 310 nM T51426 C56PRA 44574364 EC50 = 450 nM T51426 C9M5OX 44574365 EC50 = 48 nM T51426 C5M9NI 44574366 EC50 = 17 nM T51426 CZ6B9K 44577637 EC50 = 189050 nM T51426 C95BEX 44588756 EC50 = 4790 nM T51426 C8G0FP 44588757 EC50 = 6920 nM T51426 CF0OG6 44588758 EC50 = 2040 nM T51426 CB95YZ 44588759 EC50 = 5370 nM T51426 CNH0P4 44588808 EC50 = 2400 nM T51426 C13ZSU 44588809 EC50 = 3980 nM T51426 C1AP9B 44588908 EC50 = 3310 nM T51426 C8UM7P 44588909 EC50 = 6310 nM T51426 CO7W4N 44588940 EC50 = 4270 nM T51426 C2YX6O 44605418 EC50 > 100000 nM T51426 CMO1Z6 44631854 EC50 = 88 nM T51426 CS38IE 45103515 EC50 = 1121 nM T51426 C6GFZ1 45103516 EC50 = 796 nM T51426 CKI74D 45103517 EC50 = 1023 nM T51426 C4XAC1 45103619 EC50 = 99 nM T51426 CW81NZ 45103623 EC50 = 602 nM T51426 CR6DN7 45103625 EC50 = 342 nM T51426 COYU63 45104530 EC50 = 1579 nM T51426 C3JE0Z 45104531 EC50 = 368 nM T51426 CL0X4F 45104532 EC50 = 534 nM T51426 CH01QG 45104533 EC50 = 340 nM T51426 C4T7HQ 45104534 EC50 = 23 nM T51426 CH54JU 45104636 EC50 = 447 nM T51426 C4G7PQ 45104756 EC50 = 101 nM T51426 C73ATL 45104757 EC50 = 1066 nM T51426 CQC38A 45104851 EC50 = 439 nM T51426 CM7H2G 45104852 EC50 = 698 nM T51426 CBYP45 45104853 EC50 = 249 nM T51426 CP32RS 45104854 EC50 = 287 nM T51426 CJ03BS 45104855 EC50 = 271 nM T51426 CSH0P1 45104949 EC50 = 362 nM T51426 CJ30FY 45104950 EC50 = 424 nM T51426 CB8A1Y 45104951 EC50 = 194 nM T51426 CK7O5S 45104952 EC50 = 1386 nM T51426 CSQ54C 45104953 EC50 = 1317 nM T51426 CWU9D6 45105050 EC50 = 894 nM T51426 CPJD95 45105051 EC50 = 855 nM T51426 C60IXM 45105052 EC50 = 2870 nM T51426 C6C1ET 45105053 EC50 = 617 nM T51426 CR12ZK 45105054 EC50 = 1603 nM T51426 C1GZV8 45483944 EC50 = 11800 nM T51426 CDO90F 45484781 EC50 = 1300 nM T51426 COEA08 45484782 EC50 = 640 nM T51426 C2DKG6 45484804 EC50 = 1900 nM T51426 C0X1KA 45484805 EC50 = 5700 nM T51426 CV76PM 45484832 EC50 = 1300 nM T51426 C69REH 45484837 EC50 = 2700 nM T51426 CUC8Y0 45484838 EC50 = 4100 nM T51426 C2XI5K 45484845 EC50 = 3300 nM T51426 C7E3WS 45600231 EC50 = 280 nM T51426 CD3HM9 45754043 EC50 = 3800 nM T51426 CB71TA 49837867 EC50 = 500 nM T51426 CZQC64 49837869 EC50 = 300 nM T51426 CVNA15 49837870 IC50 = 50 nM T51426 CRBQ21 49837871 EC50 = 1400 nM T51426 CB1L4H 49862120 EC50 = 208 nM T51426 CK1L2C 49862121 EC50 = 385 nM T51426 C31VPM 49862122 EC50 = 365 nM T51426 C8HXF5 49862163 EC50 = 433 nM T51426 CEN0H5 49862164 EC50 = 89 nM T51426 CZV05Q 49862165 EC50 = 147 nM T51426 C01DMJ 49862166 EC50 = 225 nM T51426 C85OSV 49862205 EC50 = 101 nM T51426 C5QP3D 49862206 EC50 = 16 nM T51426 CEOA12 49862207 EC50 = 6 nM T51426 CZ90QH 49862208 EC50 = 11 nM T51426 CR8TE6 49862209 EC50 = 19 nM T51426 C8V5UA 49862247 EC50 = 155 nM T51426 CUD91T 49862248 EC50 = 2 nM T51426 C17JPF 49862249 EC50 = 20 nM T51426 CI6C5V 49862250 EC50 = 36 nM T51426 CNSG67 49862251 EC50 = 14 nM T51426 CKF8L5 49862252 EC50 = 113 nM T51426 CZ8R3B 49862294 EC50 = 107 nM T51426 CL0P8J 49862295 EC50 = 61 nM T51426 CPW46M 49862296 EC50 = 101 nM T51426 C3Q4AJ 49862297 EC50 = 179 nM T51426 CUR4C7 49862347 EC50 = 434 nM T51426 CH3AC8 49862348 EC50 = 33 nM T51426 C5I4OW 49862349 EC50 = 38 nM T51426 C08CZE 49862413 EC50 = 58 nM T51426 CVO1N4 49862414 EC50 = 189 nM T51426 CF4LH1 50905021 EC50 = 18 nM T51426 C2GTE4 50938548 IC50 = 13 nM T51426 CRH6S3 50942927 EC50 = 32 nM T51426 CR7W4O 50943000 EC50 = 111 nM T51426 CSU2P9 50943001 EC50 = 57 nM T51426 C1B2FA 50943075 EC50 = 13 nM T51426 CC8VN1 50943076 EC50 = 44 nM T51426 C9A7XD 50943077 EC50 = 76 nM T51426 CC30VJ 50943145 EC50 = 6 nM T51426 C9GTD5 50943149 EC50 = 150 nM T51426 C80TWF 50993673 IC50 = 3900 nM T51426 CK94JA 50993746 IC50 = 1500 nM T51426 C6TF7N 50993747 IC50 = 2500 nM T51426 CUB43C 51003424 IC50 = 9000 nM T51426 CF4IH7 51003425 IC50 = 17000 nM T51426 CZCL62 51003543 IC50 = 5900 nM T51426 CTJ28K 52918135 EC50 = 600 nM T51426 C6NR7I 52942081 EC50 > 10000 nM T51426 C1-MAY-02 53317017 IC50 = 210 nM T51426 CPH9I4 53317366 IC50 = 1250 nM T51426 CK6Z0H 53317477 EC50 = 140 nM T51426 CU8ZG9 53317478 EC50 = 51 nM T51426 CK5F2U 53317479 EC50 = 17 nM T51426 CSRJ76 53317508 IC50 = 14780 nM T51426 CBS0N3 53317531 EC50 = 190 nM T51426 CK27PC 53317643 EC50 = 300 nM T51426 CTN7Z0 53318647 IC50 = 12440 nM T51426 CZ4SY0 53318648 IC50 = 25120 nM T51426 C5DA1N 53318649 IC50 = 3610 nM T51426 CIG23K 53318758 EC50 = 110 nM T51426 CO0I8E 53318819 EC50 = 77 nM T51426 CTA23R 53319654 IC50 = 9 nM T51426 CB2EG3 53319655 EC50 = 5000 nM T51426 C9P4EI 53320077 EC50 = 150 nM T51426 CM6PX5 53320952 IC50 = 1300 nM T51426 CDO34E 53320953 EC50 = 50 nM T51426 CB0SR3 53320954 IC50 = 740 nM T51426 CX48PQ 53320955 EC50 = 1100 nM T51426 C14CUV 53321277 IC50 = 150 nM T51426 CHK70J 53321278 IC50 = 450 nM T51426 C9BA0Q 53321388 EC50 = 360 nM T51426 CQD07B 53321389 EC50 = 38 nM T51426 CJQ59G 53321390 EC50 = 32 nM T51426 CMH54U 53322279 EC50 = 2700 nM T51426 CLOH98 53322280 IC50 = 3900 nM T51426 CK7FI5 53322281 IC50 = 200 nM T51426 C03IST 53322282 IC50 = 3100 nM T51426 C8PV0S 53322596 IC50 = 2720 nM T51426 CM2D8W 53322704 EC50 = 52 nM T51426 CFCU21 53322705 EC50 = 24 nM T51426 C5KG8N 53322916 IC50 = 30440 nM T51426 CR57HN 53323639 EC50 = 50 nM T51426 COG20B 53323640 IC50 = 320 nM T51426 CC78EY 53323935 IC50 = 5170 nM T51426 CNP9Q2 53324081 EC50 = 340 nM T51426 CC08MY 53324265 EC50 = 90 nM T51426 CF02YQ 53324921 EC50 = 1100 nM T51426 CW82YO 53324922 EC50 = 9700 nM T51426 CGCF07 53325217 IC50 = 910 nM T51426 CX3LE0 53325218 IC50 = 3710 nM T51426 C34WXD 53325219 IC50 = 6190 nM T51426 C3B1JI 53325355 EC50 = 44 nM T51426 C8CNF4 53325356 EC50 = 14 nM T51426 CN1W4O 53325357 EC50 = 14 nM T51426 CIBV36 53325358 EC50 = 22 nM T51426 CTX07B 53325359 EC50 = 78 nM T51426 CKAI56 53325376 IC50 = 5720 nM T51426 CZX5C2 53326210 EC50 = 36 nM T51426 CL7WE2 53326211 EC50 = 9900 nM T51426 C2KSN5 53326212 EC50 = 10400 nM T51426 C28HNA 53326213 EC50 = 300 nM T51426 C41TKW 53326505 IC50 = 3800 nM T51426 C51DLX 53326892 EC50 = 200 nM T51426 C9H5YE 53361128 EC50 > 10000 nM T51426 C50BMI 53484102 EC50 = 24000 nM T51426 C49KBY 54586161 EC50 = 150 nM T51426 C6ARD5 56673082 EC50 = 500 nM T51426 CRU6B3 57389529 EC50 = 19 nM T51426 CB4Q8E 57389689 EC50 = 66 nM T51426 CYKZ60 57389849 EC50 = 8.3 nM T51426 CSF9N8 57389927 EC50 = 31 nM T51426 C1H9MK 57390008 EC50 = 4.2 nM T51426 COKE29 57652736 EC50 = 35 nM T51426 CQK0N6 59053603 EC50 = 0.42 nM T51426 CX1O9J 59053604 EC50 = 0.54 nM T51426 C7NA3K 59053728 EC50 = 0.2 nM T51426 CDJT14 59053730 EC50 = 0.46 nM T51426 C3OP5S 62715191 IC50 = 580 nM T51426 CP34ZE 62925494 EC50 = 220 nM T51426 C39PGR 62925495 EC50 = 7.2 nM T51426 C2ENA3 66927383 EC50 = 10 nM T51426 CX4PA3 67985349 EC50 = 0.27 nM T51426 CET96L 68081599 EC50 = 0.49 nM T51426 CJO65Q 68204751 EC50 = 90 nM T51426 CAZM23 68329420 EC50 = 44 nM T51426 CK6FY9 70682209 EC50 > 100000 nM T51426 C7OQ1W 70682210 EC50 = 11500 nM T51426 C78ECK 70683284 EC50 = 2600 nM T51426 CC7G2Y 70683808 EC50 = 410 nM T51426 CG3N5L 70684311 EC50 = 55000 nM T51426 CFSI97 70686469 EC50 = 22000 nM T51426 C29VEZ 70687531 EC50 = 1100 nM T51426 C76ZWP 70692259 EC50 > 10000 nM T51426 COTW72 70695911 EC50 = 3000 nM T51426 CHK95W 71205431 EC50 = 25 nM T51426 C8EOJ1 71205438 EC50 = 19 nM T51426 CIYQ62 71205440 EC50 = 9 nM T51426 CUF1R0 71228840 EC50 = 24 nM T51426 CUL7Q3 71228848 EC50 = 7 nM T51426 CR1E6Z 71228849 EC50 = 54 nM T51426 CF90MT 71228883 EC50 = 15 nM T51426 CXV96H 71456686 EC50 = 94 nM T51426 C67ZSQ 71540073 IC50 > 10000 nM T51426 C2N5WV 71599441 EC50 > 50118.72 nM T51426 CXK08C 71612420 EC50 = 6100 nM T51426 C1DR8E 71622396 EC50 = 2400 nM T51426 C58NVG 71660821 EC50 > 50118.72 nM T51426 C0VB3I 71681688 EC50 = 25000 nM T51426 CWF58U 71682019 EC50 = 30000 nM T51426 CMK58A 71722303 EC50 = 550 nM T51426 CMZ85K 72722807 EC50 = 3000 nM T51426 C2BQO3 72722945 EC50 = 1000 nM T51426 C6UWO5 74762670 EC50 > 10000 nM T51426 C0B8MV 75412552 EC50 = 15310 nM T51426 CJXG25 76284182 EC50 > 10000 nM T51426 C2H5YV 76310491 IC50 = 1100 nM T51426 CRU27S 76310492 IC50 = 3500 nM T51426 CWT02M 76310822 EC50 = 15100 nM T51426 CR0V8F 76310823 EC50 = 25290 nM T51426 C6FA7P 76311377 EC50 > 30000 nM T51426 C7O0XW 76311393 EC50 = 61150 nM T51426 CQM93B 76311394 EC50 = 14730 nM T51426 C0LE9Q 76314146 IC50 = 1200 nM T51426 C1FB2J 76314147 IC50 = 8600 nM T51426 CQVJ74 76314148 IC50 = 5400 nM T51426 CD2GS6 76314149 IC50 = 1500 nM T51426 C12DSC 76314150 IC50 = 8700 nM T51426 C39KMZ 76314443 EC50 = 24090 nM T51426 CDH8G2 76314980 EC50 = 10230 nM T51426 CELV56 76314981 EC50 = 480 nM T51426 CS7Z9N 76314982 EC50 = 790 nM T51426 C6WT0P 76314983 EC50 = 590 nM T51426 C7Y9FD 76314997 EC50 = 1210 nM T51426 C17RHY 76317717 IC50 = 5500 nM T51426 CC7W1H 76317718 IC50 = 3300 nM T51426 CE9V1T 76317719 IC50 = 25200 nM T51426 CFI1Y2 76318616 EC50 > 30000 nM T51426 CZ1JT6 76318617 EC50 = 9680 nM T51426 C0C4MB 76318618 EC50 > 30000 nM T51426 CDUP17 76318643 EC50 = 15110 nM T51426 C41FDT 76322264 EC50 = 42700 nM T51426 C5B2TR 76322265 EC50 = 2430 nM T51426 COL2Y0 76325022 IC50 = 3100 nM T51426 CV26TJ 76325023 IC50 = 5800 nM T51426 CQ05VW 76325905 EC50 = 1110 nM T51426 CF6PR5 76325918 EC50 > 30000 nM T51426 C7GR4E 76325927 EC50 = 2720 nM T51426 C5WNJ9 76328594 IC50 = 7800 nM T51426 CA4VO6 76329475 EC50 = 540 nM T51426 CZ94BJ 76329476 EC50 = 15620 nM T51426 CC2FT4 76329477 EC50 = 5990 nM T51426 C6F7RA 76329478 EC50 > 30000 nM T51426 C2UH9K 76329496 EC50 = 2500 nM T51426 CXOY63 76329502 EC50 = 13200 nM T51426 CDN9A0 76329503 EC50 = 410 nM T51426 CR9Q4F 76332274 IC50 = 1700 nM T51426 CQ70UO 76332275 IC50 = 8500 nM T51426 C3N5FV 76333117 EC50 = 4550 nM T51426 CGDF21 76333119 EC50 = 600 nM T51426 C9J0OA 76333146 EC50 = 1140 nM T51426 CY8M7G 76335912 IC50 = 2900 nM T51426 CRP5D0 76335913 IC50 = 8400 nM T51426 CTI09H 76335914 IC50 = 3200 nM T51426 C3D8ME 76336194 EC50 = 34190 nM T51426 C1BYO5 76336731 EC50 = 750 nM T51426 C5WTL8 76336749 EC50 = 1220 nM T51426 CU27JT 76336750 EC50 = 33180 nM T51426 CKT6Y5 76336751 EC50 = 7110 nM T51426 C6H4AE 76336752 EC50 = 1480 nM T51426 C9DI1A 81567254 IC50 > 100000 nM T51426 CLY2O4 84422330 EC50 = 340 nM T51426 CJY2M4 84425006 EC50 = 170 nM T51426 C6X5MD 86279340 EC50 = 1500 nM T51426 CBI06J 86346645 EC50 > 10000 nM T51426 C5VCM4 86690644 EC50 > 10000 nM T51426 CGFW70 86690646 EC50 > 10000 nM T51426 C40LQX 89405858 IC50 = 18200 nM T51426 C1JOZ9 89501446 EC50 = 6400 nM T51426 C5MOV2 89659415 EC50 > 10000 nM T51426 C7E5RV 90200534 EC50 > 10000 nM T51426 CQ78PX 90655903 EC50 = 1000 nM T51426 CRH5L1 90656005 EC50 = 4400 nM T51426 CI2Q9P 90656006 EC50 = 1000 nM T51426 C7ZDQ4 90656007 EC50 = 1300 nM T51426 CIC0M5 90656008 EC50 = 3100 nM T51426 CQK8E7 90656009 EC50 = 5800 nM T51426 C3OS1V 90656010 EC50 = 2500 nM T51426 CD79FV 90656011 EC50 = 8550 nM T51426 C0GK9L 90656012 EC50 = 720 nM T51426 CE16TD 90656013 EC50 = 7100 nM T51426 CY59UG 90656014 EC50 = 8300 nM T51426 CHNE31 90656808 IC50 = 18.4 nM T51426 CJOY36 90656809 IC50 = 130.3 nM T51426 C1SO4I 90656810 IC50 = 199.4 nM T51426 CAP4D5 90656811 IC50 = 3490 nM T51426 C9KV2R 90656812 IC50 = 1240 nM T51426 C3H4PQ 90656813 IC50 = 77.5 nM T51426 CP7R5B 90656814 IC50 = 30.9 nM T51426 C3RC6E 90656815 IC50 = 3420 nM T51426 CBPH83 90656816 IC50 = 389.5 nM T51426 C3HT5B 90656817 IC50 = 489.4 nM T51426 CZ51WS 90656818 IC50 = 5330 nM T51426 CO78EU 90656819 IC50 = 3810 nM T51426 C5UTS9 90656820 IC50 = 2040 nM T51426 CV5T8U 90656821 IC50 = 2310 nM T51426 CF48LC 90656822 IC50 = 24.3 nM T51426 CJY08E 90656823 IC50 = 5910 nM T51426 CF42HC 90656824 IC50 = 14.1 nM T51426 CF9YT2 90656825 IC50 = 23.9 nM T51426 CEOI73 90656826 IC50 = 17.7 nM T51426 CW0M7N 90656827 IC50 = 49.1 nM T51426 C8U0IN 90656828 IC50 = 52.5 nM T51426 CKC92J 90656829 IC50 = 10.2 nM T51426 CZWG10 90656830 IC50 = 76.9 nM T51426 C4S1DT 90656831 IC50 = 7.5 nM T51426 C0Z8WL 90767009 EC50 = 1590 nM T51426 CI92WR 91664317 EC50 > 10000 nM T51426 CIA15W 91754483 EC50 = 47 nM T51426 CTCN23 100941986 EC50 = 20150 nM T51426 C8QP7T 101661274 EC50 = 110 nM T51426 C0BSC7 101680019 EC50 = 8000 nM T51426 C6X3UY 101680020 EC50 = 76000 nM T51426 CP2HW1 101680021 EC50 = 91500 nM T51426 C7R6IK 101882290 EC50 = 8 nM T51426 C32OBL 101886303 EC50 = 9000 nM T51426 CC3PM5 101886309 EC50 = 2000 nM T51426 CCW4S0 101896435 EC50 = 45 nM T51426 CA6I4Y 101896436 EC50 = 700 nM T51426 CFCE51 101896437 EC50 = 2500 nM T51426 C8CJR5 102004339 EC50 > 100000 nM T51426 CQF04P 102004721 EC50 = 8900 nM T51426 CM09SC 102004737 EC50 = 5660 nM T51426 C0YXR4 102004738 EC50 = 4740 nM T51426 CIP56S 102004739 EC50 = 13300 nM T51426 C8W5NB 104900527 IC50 = 34500 nM T51426 C4YMF3 104914912 IC50 = 127 nM T51426 C1P2HC 105534625 EC50 = 100 nM T51426 C5DE6H 108745395 EC50 = 1700 nM T51426 CYN18Q 108884731 EC50 = 3800 nM T51426 C5H4JX 108933742 EC50 = 260 nM T51426 CI62TQ 110784491 EC50 = 3800 nM T51426 C4S9EM 117964962 EC50 > 10000 nM T51426 CS4GJ9 117964973 EC50 > 10000 nM T51426 CDXK37 117964975 EC50 > 10000 nM T51426 CN6RT8 117964978 EC50 > 10000 nM T51426 C96BSK 117964998 EC50 > 10000 nM T51426 C4HRT5 118063558 EC50 = 24 nM T51426 CDS9V6 118063583 EC50 = 6 nM T51426 CW27MY 118063735 EC50 = 7 nM T51426 CD01CA 118526849 EC50 > 10000 nM T51426 CT4RD5 118714597 EC50 = 280 nM T51426 C9M7RL 118714598 EC50 = 6900 nM T51426 C49HBU 118714599 EC50 = 3700 nM T51426 C5U4QT 118714600 EC50 = 10000 nM T51426 CYL4V7 118714602 EC50 = 4900 nM T51426 CN4PU6 118714603 EC50 = 5000 nM T51426 CWBF73 118714616 EC50 = 5200 nM T51426 CLZ49Y 118714617 EC50 = 480 nM T51426 CJW4A5 118714618 EC50 = 380 nM T51426 C4O7HQ 118714619 EC50 = 200 nM T51426 CDO4Q6 118714620 EC50 = 2900 nM T51426 C0R1XV 118714621 EC50 = 70 nM T51426 CV20MQ 118714622 EC50 = 71 nM T51426 CA1RT3 118714624 EC50 = 420 nM T51426 C8AS1X 118714625 EC50 = 60 nM T51426 CGI3J6 118714626 EC50 = 42 nM T51426 CB27OT 118714627 EC50 = 4700 nM T51426 CP10TG 118714628 EC50 = 480 nM T51426 C98ILP 118714629 EC50 = 1100 nM T51426 C0X3NL 118714630 EC50 = 47 nM T51426 C7KS6D 118714631 EC50 = 280 nM T51426 CR7I1H 118714632 EC50 = 150 nM T51426 CL1VI2 118714636 IC50 = 12300 nM T51426 CNA46V 118714637 EC50 = 47 nM T51426 C0ZG9J 118714638 IC50 = 15100 nM T51426 CB15VJ 118714640 EC50 = 61 nM T51426 CCQS50 118714641 EC50 = 48 nM T51426 CRGY82 118714642 EC50 = 110 nM T51426 CIV37E 118714643 EC50 = 87 nM T51426 CIP10E 118714644 EC50 = 43 nM T51426 CUEW81 118722181 EC50 = 54 nM T51426 C48GSW 118722182 EC50 = 35 nM T51426 C1IT4D 118722183 EC50 = 1230 nM T51426 CKBN73 118722184 EC50 = 309 nM T51426 CC59MO 118722185 EC50 = 617 nM T51426 CB9Q2Z 118722186 EC50 = 123 nM T51426 C2BL4J 118722187 EC50 = 20 nM T51426 CBZ75K 118724654 EC50 > 10000 nM T51426 CZP8E7 118725344 EC50 = 3400 nM T51426 CKC50A 118725345 EC50 = 2100 nM T51426 C5ENC7 118725346 EC50 = 2600 nM T51426 CTH73Y 118725347 EC50 = 2300 nM T51426 CQ4OY5 118725348 EC50 = 8500 nM T51426 C9M1BC 118725349 EC50 = 7000 nM T51426 C4PZF0 119218407 IC50 = 102 nM T51426 CE9H7Y 121322331 EC50 = 50 nM T51426 C2VU7H 121322333 EC50 = 290 nM T51426 C6TBD2 121345502 EC50 > 20000 nM T51426 CB6A8H 121355127 EC50 = 60 nM T51426 CGR82H 121369761 EC50 = 230 nM T51426 CDCL54 121425568 EC50 = 230 nM T51426 C19HXR 121428806 EC50 = 470 nM T51426 CG9U3D 122188872 IC50 > 100000 nM T51426 C06NSD 122188980 IC50 > 100000 nM T51426 C49IQH 122188981 IC50 = 12700 nM T51426 CYR3P8 122188982 IC50 = 8800 nM T51426 CU79EV 122188983 IC50 = 5900 nM T51426 C4SPZ2 122188984 IC50 = 34200 nM T51426 CE51BK 122188985 IC50 = 7200 nM T51426 CBIF13 122188986 IC50 = 600 nM T51426 C9Y0DX 122188987 IC50 = 13600 nM T51426 CEXP96 122188988 IC50 > 100000 nM T51426 C1BDF9 122188989 IC50 > 100000 nM T51426 CZX3V8 122188990 IC50 > 100000 nM T51426 CP4AS0 122188991 IC50 > 100000 nM T51426 CB03HG 122188992 IC50 > 100000 nM T51426 C7L5ES 122188993 IC50 = 15500 nM T51426 CM0I6F 122188994 IC50 = 5200 nM T51426 C8VE9N 122188995 IC50 = 3600 nM T51426 CX2UI3 122188996 IC50 = 9800 nM T51426 CR49WV 122188997 IC50 = 8600 nM T51426 C64TDG 122188998 IC50 = 13900 nM T51426 C2YKU6 122188999 IC50 = 28700 nM T51426 CSZO56 122189000 IC50 = 5000 nM T51426 C36CJK 122189001 IC50 = 2500 nM T51426 CIP8J6 122189002 IC50 = 1400 nM T51426 CFS35K 122189003 IC50 > 100000 nM T51426 C9P6XW 122189004 IC50 > 100000 nM T51426 CHE9T4 122189005 IC50 > 100000 nM T51426 CS8RF4 122189006 IC50 = 3900 nM T51426 CQX0Z5 122189007 IC50 = 6300 nM T51426 C7OPK0 122189008 IC50 > 100000 nM T51426 CF37GP 122189009 IC50 > 100000 nM T51426 CRY8N5 122190169 EC50 = 4200 nM T51426 CT9UJ0 122194860 EC50 = 15470 nM T51426 C8YQB4 122194861 EC50 = 2400 nM T51426 C7HC9N 122194862 EC50 = 12140 nM T51426 CO9ED1 122194864 EC50 = 40740 nM T51426 CIM52E 122194865 EC50 = 940 nM T51426 C3O7RZ 122194866 EC50 = 3030 nM T51426 CYQV03 122194867 EC50 = 64890 nM T51426 C9Y8FR 122194868 EC50 = 140 nM T51426 CJ0G1P 122194869 EC50 = 10400 nM T51426 C21VJS 122194870 EC50 = 5640 nM T51426 C4NWA6 122194871 EC50 = 20240 nM T51426 CZM8O4 122194873 EC50 = 3360 nM T51426 CRAS43 122201312 EC50 = 230 nM T51426 C53XOE 122657467 EC50 = 71 nM T51426 C9OX2H 122657470 EC50 = 145 nM T51426 CUG35B 122657481 EC50 = 520 nM T51426 CA6D2C 122657485 EC50 = 480 nM T51426 CAP93M 122657488 EC50 = 38 nM T51426 C1LOI7 122657494 EC50 = 16 nM T51426 CT82OU 122657507 EC50 = 23 nM T51426 C39HNL 122657530 EC50 = 150 nM T51426 CSIH39 122657534 EC50 = 13 nM T51426 CW4F8P 122657541 EC50 = 25 nM T51426 C0XWI7 127029952 EC50 = 11000 nM T51426 CMWK92 127040472 EC50 = 15390 nM T51426 C45QST 127040473 EC50 = 29940 nM T51426 CZH28N 127048817 EC50 = 220 nM T51426 C05GLD 127048818 EC50 = 373 nM T51426 CJ7M0E 127049120 EC50 = 15 nM T51426 C6JMY2 127052365 EC50 = 4 nM T51426 CZTI57 127052669 EC50 = 44 nM T51426 C1HO8B 127052968 EC50 = 79 nM T51426 CTV6J3 129315293 EC50 = 400 nM T51426 CXUK13 130261792 IC50 = 1250 nM T51426 CA2U8G 132210217 EC50 = 2.6 nM T51426 CSED10 132210223 EC50 = 3.4 nM T51426 C07LVG 132210228 EC50 = 4.5 nM T51426 CEYF71 132210258 EC50 = 15 nM T51426 C5K4UR 132938263 IC50 = 126100 nM T51426 C1TWR2 134214576 EC50 = 1000 nM T51426 CF65AU 135385301 EC50 = 46 nM T51426 CY5TN6 135505551 EC50 = 10500 nM T51426 CJ2P7C 136206345 EC50 = 1700 nM T51426 CP4OZ2 136206346 EC50 = 1100 nM T51426 C9EOV6 136206347 EC50 = 1100 nM T51426 CQTU46 136226153 EC50 > 150000 nM T51426 C3VY2J 136226155 EC50 = 3000 nM T51426 CK8ST6 136226156 EC50 = 1300 nM T51426 C9FIK0 136226157 EC50 > 150000 nM T51426 CQ9GM3 136226158 EC50 > 150000 nM T51426 CI43SP 136226161 EC50 > 150000 nM T51426 CHPT89 136226162 EC50 = 2000 nM T51426 CC07ZU 136226163 EC50 > 150000 nM T51426 C4AND7 136244210 EC50 = 2400 nM T51426 CJI54V 136244211 EC50 = 2000 nM T51426 CGW08L 136244212 EC50 = 1800 nM T51426 C8Z6CR 136244265 EC50 = 1900 nM T51426 CFQ0I6 136244266 EC50 = 3300 nM T51426 CBW13R 136254228 EC50 = 1300 nM T51426 CK0E2H 136254229 EC50 = 2700 nM T51426 CD7EQ4 136254230 EC50 = 3900 nM T51426 C35XEO 136254231 EC50 = 1900 nM T51426 CPA78C 136254232 EC50 = 2200 nM T51426 CT0L4U 136254233 EC50 = 1700 nM T51426 C1FAZ9 136254234 EC50 = 1500 nM T51426 CMVL97 136254235 EC50 = 3500 nM T51426 CS0ZV8 136254236 EC50 = 3600 nM T51426 CA51CI 136254237 EC50 = 1400 nM T51426 CF5Y2V 136254238 EC50 = 2600 nM T51426 CMZ81D 136254239 EC50 = 3500 nM T51426 CN1X5Y 136254240 EC50 = 1200 nM T51426 CGK9U8 136254241 EC50 = 1800 nM T51426 CR2U5I 136254242 EC50 = 1100 nM T51426 CTJ69N 136254243 EC50 = 990 nM T51426 C9X4EB 136254244 EC50 = 3400 nM T51426 CG29XW 136259625 EC50 = 14000 nM T51426 C5M7NR 137631417 IC50 = 3870 nM T51426 CAD2P3 137631891 EC50 = 20.4 nM T51426 CJC9V2 137631929 EC50 = 1580 nM T51426 CV1U8F 137631946 EC50 = 180 nM T51426 CNW47H 137632309 IC50 = 112900 nM T51426 CO6A5L 137632414 IC50 = 118500 nM T51426 CJV2Y3 137633688 EC50 = 76 nM T51426 C1I6AV 137633748 EC50 = 1100 nM T51426 CZ37EN 137633799 IC50 = 17300 nM T51426 CZ3WM6 137634192 EC50 = 1200 nM T51426 C0D8QN 137634352 EC50 = 1200 nM T51426 CZ4OB3 137634692 IC50 = 75300 nM T51426 CM08UD 137634906 IC50 = 28500 nM T51426 C91ALG 137636409 EC50 = 170 nM T51426 CKL1B0 137636686 EC50 = 120 nM T51426 CPDH58 137637016 IC50 = 209500 nM T51426 C1FWB9 137637324 EC50 = 750 nM T51426 CR37SG 137637968 EC50 = 7.8 nM T51426 CE2UM0 137637982 EC50 = 26 nM T51426 CT49FJ 137638497 EC50 = 460 nM T51426 C2M1FY 137639064 IC50 = 15300 nM T51426 C7I6GS 137639592 IC50 = 43400 nM T51426 CX3W4Q 137639938 EC50 = 350 nM T51426 C0VD1N 137639961 EC50 = 3200 nM T51426 C2F6GZ 137640822 EC50 = 0.4 nM T51426 C3SH9N 137641234 IC50 = 6600 nM T51426 C39SQB 137641372 EC50 = 7500 nM T51426 C5C7YN 137642545 EC50 = 3060 nM T51426 CNA45O 137643486 IC50 = 3580 nM T51426 C1F9TG 137643657 IC50 = 125500 nM T51426 C72NWG 137644140 EC50 = 14 nM T51426 CL6AF0 137644141 EC50 = 8.8 nM T51426 C25BCT 137644228 EC50 = 810 nM T51426 C6TUV0 137644316 IC50 = 417500 nM T51426 CZB24M 137644358 IC50 = 18200 nM T51426 CS96PL 137644758 EC50 = 5300 nM T51426 CF6KI8 137645153 EC50 = 1200 nM T51426 CMT46B 137645546 EC50 = 230 nM T51426 CUOH02 137645612 IC50 = 16200 nM T51426 CP5A7K 137646226 EC50 = 220 nM T51426 CSH1R5 137647356 EC50 = 430 nM T51426 CS3M4I 137647530 EC50 = 1300 nM T51426 CRG0D7 137649191 IC50 = 10400 nM T51426 C83WFZ 137649837 EC50 = 1.5 nM T51426 C09JQM 137650621 EC50 = 520 nM T51426 CNIP43 137650661 EC50 = 830 nM T51426 C09NEO 137650679 IC50 = 24400 nM T51426 CVF94A 137650876 IC50 = 35200 nM T51426 C3GIV8 137650941 EC50 = 0.3 nM T51426 CE17JZ 137651395 EC50 = 7.4 nM T51426 CB05RX 137651449 EC50 = 220 nM T51426 C7V2AU 137651579 EC50 = 200 nM T51426 C2BUF3 137651721 IC50 = 104600 nM T51426 CS2LU0 137651997 EC50 = 160 nM T51426 C0LON9 137652125 EC50 = 2000 nM T51426 CG7B2M 137652547 EC50 = 100 nM T51426 CMKJ42 137653039 IC50 = 87500 nM T51426 C7MV8K 137653251 EC50 = 730 nM T51426 CQDA52 137653334 EC50 = 830 nM T51426 CIO7P5 137653377 IC50 = 174500 nM T51426 CN7M3P 137653534 IC50 = 3980 nM T51426 CK7JD5 137653822 EC50 = 670 nM T51426 CYU7Q6 137654386 IC50 = 2560 nM T51426 CF3N9H 137654427 EC50 = 160 nM T51426 CSM10L 137654774 EC50 = 260 nM T51426 C9AL7X 137655456 IC50 = 398800 nM T51426 C70WUN 137655766 EC50 = 6400 nM T51426 CP9UJ4 137656136 EC50 = 970 nM T51426 CRNM57 137656530 EC50 = 81 nM T51426 C43HUX 137656636 EC50 = 140 nM T51426 CY71ND 137656982 IC50 = 23100 nM T51426 CG9SV5 137656992 IC50 = 8110 nM T51426 C0MRN7 137657016 IC50 = 65600 nM T51426 CE9UY7 137657030 EC50 = 80 nM T51426 C4IN0L 137658784 EC50 = 2900 nM T51426 C4GZ0V 137659284 IC50 = 102200 nM T51426 CQC98F 137659585 EC50 = 1000 nM T51426 CQTS70 137659957 EC50 = 1300 nM T51426 CS7QL1 137660000 EC50 = 16 nM T51426 CA20WB 137661482 IC50 = 77100 nM T51426 CGAY68 139051176 EC50 = 6660 nM T51426 CPW8S5 145089899 EC50 = 150 nM T51426 C6A8TR 145177795 EC50 = 20 nM T51426 CRPI59 145177799 EC50 = 1800 nM T51426 CS4FN3 145177850 EC50 = 300 nM T51426 C52EPH 145177933 EC50 = 1100 nM T51426 CSV4O1 145177998 EC50 = 700 nM T51426 CAT26W 145178037 EC50 = 2700 nM T51426 CO58SC 145178076 EC50 = 370 nM T51426 C17HLI 145948883 IC50 = 6000 nM T51426 COR8C3 145949229 EC50 = 1500 nM T51426 CMV9X3 145949320 EC50 = 130 nM T51426 CM8U0C 145949696 IC50 < 0.001 nM T51426 CPZX74 145949879 EC50 = 100 nM T51426 CQ54UR 145950045 EC50 = 300 nM T51426 C51ZYQ 145950691 EC50 = 230 nM T51426 CE3O8Q 145950705 IC50 = 17400 nM T51426 C46OIX 145954350 EC50 = 150 nM T51426 CE4B7L 145954756 EC50 = 300 nM T51426 CWM65Q 145954891 IC50 < 0.001 nM T51426 CTY36E 145955086 IC50 = 130 nM T51426 C5S9DQ 145955411 EC50 = 70 nM T51426 C1L3NH 145955827 EC50 = 80 nM T51426 CJE17T 145955983 EC50 = 600 nM T51426 CC51UX 145955988 EC50 = 30 nM T51426 CCM3K5 145955991 IC50 = 0.002 nM T51426 CK82JA 145956106 IC50 = 0.8 nM T51426 CYS2J3 145956445 EC50 = 80 nM T51426 C0U1NG 145956850 EC50 = 110 nM T51426 CT0S9O 145956999 IC50 = 0.06 nM T51426 CD3L4I 145957112 IC50 = 1300 nM T51426 CRU2G4 145957191 IC50 = 4510 nM T51426 CA85XR 145957205 EC50 = 80 nM T51426 CQ15RN 145957458 IC50 = 0.006 nM T51426 CE4S6X 145957828 EC50 = 300 nM T51426 C6OZ8N 145959237 EC50 = 280 nM T51426 C86EZG 145959438 EC50 = 110 nM T51426 C1LQ5R 145972671 IC50 = 1 nM T51426 C7GN5U 145972897 EC50 = 300 nM T51426 CA6U8M 145973129 EC50 = 30 nM T51426 C0DEA1 145974037 EC50 > 50118.72 nM T51426 C65FXH 145974346 EC50 = 240 nM T51426 C6R0LB 145982508 IC50 = 5000 nM T51426 C2AD3K 145982631 IC50 = 80 nM T51426 C9ELC6 145982776 IC50 = 1.3 nM T51426 CA7L4Y 145982794 IC50 = 700 nM T51426 C4X9VB 145982813 IC50 = 3700 nM T51426 C1MV7G 145983817 IC50 = 140 nM T51426 C5O8AF 145983875 IC50 = 190 nM T51426 CT1Z9K 145983940 IC50 = 9100 nM T51426 C1J9EV 145984224 IC50 = 2200 nM T51426 C7QB6J 145984308 IC50 = 8100 nM T51426 CW0X7R 145984832 IC50 = 3300 nM T51426 C92HDJ 145985373 IC50 = 1500 nM T51426 C1OBY6 145985915 IC50 = 280 nM T51426 CCM06Y 145985943 IC50 = 170 nM T51426 CV9RF4 145986225 IC50 = 220 nM T51426 CSQ32X 146302376 EC50 = 2060 nM T51426 CW4UE1 146302377 EC50 = 2800 nM T51426 C4IHF5 146302381 EC50 = 6670 nM T51426 CA84PG 146311945 EC50 = 2930 nM T51426 CQEC78 146311962 EC50 = 830 nM T51426 C7IMJ9 146311964 EC50 = 4370 nM T51426 CUZN97 150026820 IC50 = 40400 nM T51426 CFQB04 150277481 EC50 = 460 nM T51426 CUXJ27 150353286 EC50 = 5400 nM T51426 CNXC41 150485180 EC50 = 740 nM T51426 CI06GK 150542873 EC50 = 670 nM T51426 CK19ZP 150793526 EC50 = 19740 nM T51426 CB81KT 150824883 EC50 = 1400 nM T51426 CY87HN 150979017 EC50 = 810 nM T51426 C81URY 151002530 EC50 = 1090 nM T51426 C41TZM 151011965 IC50 = 25700 nM T51426 CR51CE 151189666 EC50 = 940 nM T51426 CCB21Z 151228499 IC50 = 1170 nM T51426 C48NGU 151595152 EC50 = 10170 nM T51426 C9PXK3 152221886 EC50 = 300 nM T51426 C4V6HL 155510835 IC50 = 1101 nM T51426 C3K4GJ 155511574 EC50 > 10000 nM T51426 CBE26Q 155511678 EC50 = 30080 nM T51426 CKRM42 155511689 EC50 = 14700 nM T51426 C5NYV8 155512376 EC50 = 3340 nM T51426 C3MR9Y 155512726 EC50 = 10190 nM T51426 CGFO69 155515061 EC50 = 2170 nM T51426 CQ4IX9 155515717 EC50 = 20250 nM T51426 C1YPS3 155516251 EC50 = 2230 nM T51426 CH5AP2 155519174 EC50 = 55490 nM T51426 CIV9S4 155519410 EC50 = 20320 nM T51426 C29YMN 155519456 EC50 = 2580 nM T51426 C96WRT 155519615 EC50 = 2300 nM T51426 C5JB3I 155520144 EC50 > 10000 nM T51426 CZC52H 155520474 EC50 = 17600 nM T51426 CB4XF3 155520673 EC50 = 8800 nM T51426 C3GX0D 155521423 EC50 = 9620 nM T51426 C7BOM5 155522755 IC50 = 35 nM T51426 C2YK4C 155523003 IC50 = 781 nM T51426 C8QA3I 155523525 EC50 = 50250 nM T51426 CB8PU3 155523526 IC50 = 59.8 nM T51426 CR48MT 155524690 IC50 < 20000 nM T51426 CE7GJ5 155525365 EC50 = 730 nM T51426 CP4A7L 155525439 EC50 = 16680 nM T51426 CP16TI 155526101 IC50 = 33800 nM T51426 CJ79QA 155527087 EC50 = 430 nM T51426 CF8N4M 155527188 EC50 = 2520 nM T51426 CBCM58 155528505 IC50 = 81 nM T51426 CIP92H 155529056 IC50 < 20000 nM T51426 CONH95 155529489 EC50 = 15470 nM T51426 C3CGD2 155529590 IC50 = 41 nM T51426 C3MBZ9 155529962 IC50 = 28400 nM T51426 CY0N8B 155530924 EC50 > 10000 nM T51426 CAE41I 155531534 EC50 = 4690 nM T51426 CD2OJ6 155531556 EC50 = 5600 nM T51426 CA3I8D 155531998 EC50 = 24480 nM T51426 CIY2S1 155532027 IC50 = 550 nM T51426 C1LED9 155534516 EC50 > 10000 nM T51426 C63HSA 155534748 IC50 > 50000 nM T51426 CJP4C9 155535302 EC50 = 90 nM T51426 CG0I5O 155535307 IC50 < 20000 nM T51426 C1E3ZA 155535937 IC50 = 18.3 nM T51426 CGX5I9 155535971 IC50 = 550 nM T51426 C2Q9NZ 155536161 EC50 = 2700 nM T51426 CTNM57 155536707 EC50 = 10970 nM T51426 CQ78WP 155536938 EC50 = 12070 nM T51426 CFHG51 155537881 EC50 = 16430 nM T51426 CT96GK 155538233 IC50 = 859 nM T51426 CRL8F5 155538318 IC50 = 550 nM T51426 COP7X8 155539171 IC50 > 10000 nM T51426 CNB1R8 155539608 EC50 = 11860 nM T51426 CU9JO2 155540517 EC50 > 10000 nM T51426 CH28PV 155540571 EC50 = 14380 nM T51426 CR6JV4 155540812 EC50 = 4300 nM T51426 CU3PG2 155541129 IC50 = 27300 nM T51426 CP73ED 155541638 IC50 = 7000 nM T51426 CUK6D0 155541843 IC50 = 2.4 nM T51426 C14XBT 155544762 EC50 > 10000 nM T51426 C84OYC 155546534 EC50 = 1150 nM T51426 CF5J6L 155547555 IC50 = 799 nM T51426 C5L8AS 155548009 EC50 = 3590 nM T51426 C3MA6N 155548163 EC50 = 290 nM T51426 C7EY2U 155549961 IC50 = 27000 nM T51426 CW8O6X 155550231 EC50 = 17500 nM T51426 CXJS46 155550548 EC50 = 12430 nM T51426 CPE6Y8 155551587 IC50 = 10500 nM T51426 CY5N6P 155554675 EC50 = 1260 nM T51426 CQJ1U7 155556426 IC50 < 0.001 nM T51426 C1SGZ3 155556810 EC50 = 38160 nM T51426 C1MT2Z 155557091 IC50 = 978 nM T51426 CNW3I0 155557101 IC50 = 9.3 nM T51426 CV8R5M 155557882 EC50 = 2840 nM T51426 CEYB64 155558519 EC50 = 46960 nM T51426 C4B9MQ 155558781 IC50 = 20500 nM T51426 CE76GZ 155560459 IC50 < 0.001 nM T51426 CKC12Q 155560821 EC50 = 120 nM T51426 CI9CT3 155561761 IC50 = 38700 nM T51426 CV79NJ 155562422 EC50 = 7320 nM T51426 CQB30N 155564258 IC50 = 23000 nM T51426 C60UTW 155564605 EC50 = 13260 nM T51426 C8WQ5Z 155567289 EC50 = 520 nM T51426 CCO64L 155567642 EC50 = 6000 nM T51426 CY5HJ8 155569012 IC50 = 53 nM T51426 D00TFA 3392731 IC50 = 4910 nM T51426 D01GUG 24178658 IC50 = 2400 nM T51426 D01MYO 5326713 EC50 = 25 nM T51426 D02YJL 387316 EC50 = 3000 nM T51426 D04KWH 176157 IC50 = 2770 nM T51426 D04SEX 446849 IC50 = 1310 nM T51426 D0B5FC 447912 EC50 = 1000 nM T51426 D0B7AH 45483949 EC50 > 100000 nM T51426 D0D8IS 12544 EC50 = 3000 nM T51426 D0G9YL 16214849 EC50 = 68 nM T99840 D00GPQ 46224413 IC50 = 1.2 nM T99840 D01LXD 9843750 IC50 = 38 nM T99840 D02HNG 9803433 IC50 = 5 nM T99840 D02JOH 46883536 IC50 = 0.13 nM T99840 D03MFQ 9996409 IC50 = 40000 nM T99840 D05FGR 92337 IC50 = 307000 nM T99840 D09ZVC 11269353 IC50 = 1.6 nM T99840 D0EV5O 46853593 EC50 = 29 nM T99840 D0F0JJ 11560787 IC50 = 64 nM T99840 D0I1OS 46854987 EC50 = 17 nM T99840 D0I3WC 49867930 IC50 = 4 nM T99840 D0O8UB 53241828 IC50 = 30 nM T99840 D0XI4P 91844660 IC50 = 7 nM T99840 D0D8IZ 25159185 IC50 = 8 nM T99840 D0K2YO 11964527 IC50 = 50 nM T99840 C40BXC 3803 IC50 = 30000 nM T99840 C19WAN 92803 EC50 = 5700 nM T99840 CA5BV8 169545 IC50 = 900 nM T99840 CQL19V 822847 IC50 = 1004 nM T99840 C5CG7L 965266 IC50 > 30000 nM T99840 CM73HW 2338583 IC50 > 40000 nM T99840 COK1Y6 2470340 IC50 > 40000 nM T99840 C0JR9A 2842595 IC50 = 2002 nM T99840 C5V6TP 3103157 IC50 = 2300 nM T99840 CK93HP 3844414 IC50 = 1540 nM T99840 C2B6AE 4788452 IC50 > 10000 nM T99840 CG5CH7 5155899 IC50 = 8278 nM T99840 C79BWF 5311272 IC50 = 500 nM T99840 CJ8P4T 5352624 IC50 = 53000 nM T99840 C0W3XG 5479543 IC50 = 17 nM T99840 CQ94WM 6324639 IC50 = 90 nM T99840 C76SLZ 7200833 IC50 = 966 nM T99840 CI8N0S 9805486 IC50 = 1 nM T99840 CPUY29 9807338 IC50 = 2.3 nM T99840 CI48QZ 9840950 IC50 = 651 nM T99840 CGSO64 9849380 IC50 = 5.6 nM T99840 C7TAZ2 9850372 IC50 = 17000 nM T99840 C3NF1M 9867067 IC50 = 0.19 nM T99840 C6KG4D 9874174 IC50 = 10 nM T99840 C0PN1K 9887090 IC50 = 491 nM T99840 CN3FH5 9893310 IC50 = 13.2 nM T99840 CIUM38 9901028 IC50 = 4408 nM T99840 C7Z5LV 9906160 IC50 = 70 nM T99840 CR91HS 9909323 IC50 = 32700 nM T99840 CHP82G 9910347 IC50 = 0.7 nM T99840 CD21QJ 9929326 IC50 = 3 nM T99840 C3KA5Q 9987560 IC50 = 70 nM T99840 COFE18 10002640 IC50 = 0.015 nM T99840 C0H1VQ 10117786 IC50 = 88 nM T99840 CWH3N7 10120043 IC50 = 56 nM T99840 C7ZR4N 10127574 IC50 = 570 nM T99840 CAQ5C6 10129054 IC50 = 8 nM T99840 CVX4J2 10143259 IC50 = 39 nM T99840 CXB8A6 10143260 IC50 = 540 nM T99840 C1M6SJ 10151615 IC50 = 6420 nM T99840 CLIO84 10163543 IC50 = 394 nM T99840 CU1A2J 10164752 IC50 = 2959 nM T99840 CG31VE 10175216 IC50 = 17 nM T99840 CR6LU7 10185072 IC50 = 299 nM T99840 CHL6W8 10194301 IC50 = 1970 nM T99840 C9MP6N 10194302 IC50 = 10620 nM T99840 CEV5A9 10196568 IC50 = 67 nM T99840 CPML95 10206761 IC50 = 504 nM T99840 C1AI8H 10227941 IC50 = 1096 nM T99840 CY7HG6 10239951 IC50 = 11 nM T99840 C2NU0D 10273953 IC50 = 4488 nM T99840 COQ19A 10277002 IC50 = 1644 nM T99840 C7FUL5 10311969 IC50 = 16 nM T99840 CG58VR 10341444 IC50 = 34200 nM T99840 C46JQA 10341445 IC50 = 24000 nM T99840 C9RE5W 10430137 IC50 = 22 nM T99840 CL3TN5 10434562 IC50 = 4.2 nM T99840 C0QNE9 10435235 EC50 = 0.119 nM T99840 CG2RL8 10459991 IC50 = 160 nM T99840 C2J6TA 10486685 IC50 = 780 nM T99840 CQ29TO 11062179 IC50 = 30000 nM T99840 CCR6J0 11152627 IC50 = 304 nM T99840 CN1L7M 11166476 IC50 = 400 nM T99840 C7LU4F 11169411 IC50 = 5000 nM T99840 C8SN4H 11169663 IC50 = 800 nM T99840 CTSQ29 11189908 IC50 = 230 nM T99840 C62ZWP 11192631 IC50 = 4000 nM T99840 C4CN2H 11193105 IC50 = 8000 nM T99840 CTP7N8 11226810 IC50 = 7000 nM T99840 CCD9V7 11240339 IC50 = 28 nM T99840 CJB5O8 11249248 IC50 = 7.1 nM T99840 CD8XH1 11250722 IC50 = 1000 nM T99840 CIDX13 11251926 IC50 = 9 nM T99840 CGZ49K 11257831 IC50 = 0.09 nM T99840 C3TV2Y 11273945 IC50 = 6000 nM T99840 C2F7MP 11285138 IC50 = 10 nM T99840 CTX52V 11297905 IC50 = 4700 nM T99840 CQ2P1S 11297908 IC50 = 26 nM T99840 CJ4R9F 11305056 IC50 = 0.024 nM T99840 CB9D7R 11306390 IC50 = 1 nM T99840 CWSA02 11319688 IC50 = 30 nM T99840 CJ6P7M 11329213 IC50 = 8.6 nM T99840 CL0GS1 11343941 IC50 = 14 nM T99840 C9LVZ8 11351105 IC50 = 3500 nM T99840 CQAS73 11366816 IC50 = 10000 nM T99840 CX8DT9 11366854 IC50 = 3100 nM T99840 C80KEI 11366911 IC50 = 910 nM T99840 C9S0MA 11376832 IC50 = 36.1 nM T99840 CHX4B9 11396006 IC50 = 0.042 nM T99840 CK3A1O 11423529 IC50 = 11000 nM T99840 CHW4L9 11430149 IC50 = 320 nM T99840 C63FEX 11431866 IC50 = 315 nM T99840 C7KLS0 11431964 IC50 = 76 nM T99840 CQ45UY 11454028 IC50 = 2.6 nM T99840 CW17SH 11456449 IC50 = 3000 nM T99840 CHZI35 11476771 IC50 = 76 nM T99840 C0TR9L 11479461 IC50 = 3000 nM T99840 C8WI9Y 11488357 IC50 = 100 nM T99840 CUO49D 11490643 IC50 = 60 nM T99840 CZ5JD8 11491881 IC50 = 16 nM T99840 CS6KW9 11494770 IC50 = 10 nM T99840 CL02TM 11503850 IC50 = 170 nM T99840 C2BI4M 11510496 IC50 = 9.1 nM T99840 CR71GB 11526691 IC50 = 9.9 nM T99840 C8YHU5 11548091 IC50 = 40 nM T99840 CR75FZ 11577204 IC50 = 15 nM T99840 C4BCJ3 11584234 IC50 = 6 nM T99840 CE9C5X 11596669 IC50 = 5 nM T99840 C6FAC1 11597267 IC50 = 80 nM T99840 CKDQ36 11627523 IC50 = 15 nM T99840 CQ75LF 11649620 IC50 = 20 nM T99840 C1ND2H 11697625 EC50 = 1258.93 nM T99840 C2LPQ8 11713496 IC50 = 120 nM T99840 C9Z6LE 11744162 IC50 = 5 nM T99840 CGTO42 11754136 IC50 = 10 nM T99840 C6Y8RF 11763616 IC50 = 800 nM T99840 CU2XG6 11815760 IC50 = 360 nM T99840 CYM80H 11817327 IC50 > 40000 nM T99840 CQ26XH 11851431 IC50 = 2.5 nM T99840 C0FSC7 11957110 IC50 = 0.06 nM T99840 C0YZH6 12147040 IC50 = 600 nM T99840 CQF06G 15071516 IC50 > 100000 nM T99840 C8WZH7 15208713 IC50 > 80000 nM T99840 C2D9TY 15344717 IC50 = 3100 nM T99840 C4VGL7 15767758 IC50 = 3000 nM T99840 CTM5I8 15942638 IC50 = 4 nM T99840 CA06DN 15953832 IC50 = 0.24 nM T99840 C6K8ZI 16035476 IC50 = 2 nM T99840 C7C2IK 16037832 IC50 = 3 nM T99840 CRT2F4 16043233 IC50 = 2.9 nM T99840 C8JZ4F 16043234 IC50 = 2000 nM T99840 CWD6X4 16045311 IC50 = 879 nM T99840 C7XPD5 16045393 IC50 = 151 nM T99840 CKOF24 16045394 IC50 = 6443 nM T99840 CSKY14 16045395 IC50 = 8 nM T99840 CWR7C1 16045555 IC50 = 26 nM T99840 CZB5M6 16085321 EC50 = 100 nM T99840 C9VPN2 16098384 EC50 = 20000 nM T99840 CCR68Z 16098385 EC50 > 20000 nM T99840 C51CIY 16098413 IC50 = 8500 nM T99840 C2WKD8 16098417 IC50 > 80000 nM T99840 CVYP36 16098434 IC50 > 40000 nM T99840 CPH4M3 16098435 IC50 = 2900 nM T99840 CP79WX 16112999 IC50 = 0.4 nM T99840 CSV24U 16655068 IC50 = 7500 nM T99840 C85AMK 16681308 IC50 = 21.2 nM T99840 CY1IH6 16722524 IC50 = 30 nM T99840 C70XVQ 16730389 IC50 = 598 nM T99840 CJ5YM2 16730390 IC50 = 80.9 nM T99840 CZW3O4 16730475 IC50 = 87 nM T99840 CAR4X1 16730476 IC50 = 5.4 nM T99840 C3XR6P 16730477 IC50 = 3.4 nM T99840 CF4LC6 16730478 IC50 = 776 nM T99840 CJ6YP9 16730566 IC50 = 536 nM T99840 C3BQ9R 16730567 IC50 = 120 nM T99840 C30OCW 16730568 IC50 = 10.2 nM T99840 CJ46CG 16730569 IC50 = 431 nM T99840 CODA06 16730724 IC50 = 244 nM T99840 CP30ZR 16730725 IC50 = 858 nM T99840 C7R1VI 16730727 IC50 > 40000 nM T99840 CC7QG9 16730799 IC50 = 350 nM T99840 C2PDT9 17747070 Ki = 2.6 nM T99840 CG3J5R 17747160 IC50 = 0.2 nM T99840 CAV2Z1 17986064 IC50 > 1000 nM T99840 C3G5ES 17986074 IC50 = 190 nM T99840 C0PRT8 17986076 IC50 = 7 nM T99840 CAN4I0 17986083 IC50 = 6000 nM T99840 C6MBD8 17986087 IC50 > 1000 nM T99840 C1RNQ6 17986094 IC50 > 1000 nM T99840 CK4RU9 17986184 IC50 = 70 nM T99840 CDC91U 18455128 IC50 = 1100 nM T99840 CVNB70 18455435 IC50 = 900 nM T99840 CLEI18 21048992 IC50 = 2.2 nM T99840 CS2EQ3 21049006 IC50 = 1.7 nM T99840 C3CL6R 21072502 IC50 = 3.3 nM T99840 C3CQZ6 21963897 IC50 = 4.2 nM T99840 CA48DB 21963931 IC50 = 1.4 nM T99840 C4YP3O 21963960 IC50 = 8.8 nM T99840 C38MFL 21963963 IC50 = 2.1 nM T99840 C6A7PO 21963967 IC50 = 21.5 nM T99840 CB18XR 21963968 IC50 = 148 nM T99840 CW3K9Z 21963972 IC50 = 14.3 nM T99840 CQH9L3 21963984 IC50 = 1.3 nM T99840 CO1UT3 21963988 IC50 = 1 nM T99840 CL74HI 22147970 IC50 = 1.65 nM T99840 C0A2BJ 22275595 IC50 = 40 nM T99840 CGF72V 22275717 IC50 = 2100 nM T99840 C15ZNF 22485769 IC50 = 510 nM T99840 C8LP1I 22984074 IC50 = 210 nM T99840 C32HUC 23028858 IC50 = 35 nM T99840 C05UKY 23509685 IC50 > 100000 nM T99840 CD6T3Z 23571062 IC50 = 0.06 nM T99840 CX1S4N 23571063 IC50 = 0.17 nM T99840 CYS7G4 23571064 IC50 = 0.42 nM T99840 C3GVY5 23571065 IC50 = 0.12 nM T99840 CU6IF5 23571066 IC50 = 0.82 nM T99840 CIBK15 23571067 IC50 = 0.08 nM T99840 C5T1SC 23571069 IC50 = 0.15 nM T99840 CXQ8R3 23571070 IC50 = 0.03 nM T99840 CC6N9Y 23571085 IC50 = 0.06 nM T99840 C68MVY 23571092 IC50 = 0.41 nM T99840 C06ZKN 23571093 IC50 = 0.06 nM T99840 CEPG49 23571096 IC50 = 0.07 nM T99840 CF7X5B 23571100 IC50 = 0.42 nM T99840 CB1R2P 23571105 IC50 = 0.34 nM T99840 C94OLI 23571205 IC50 = 0.21 nM T99840 C09CFT 23590946 IC50 = 4.7 nM T99840 CQ0JA6 23590952 IC50 = 0.51 nM T99840 CX36KQ 23627219 IC50 = 27 nM T99840 CNT92F 23656215 IC50 = 0.3 nM T99840 CIT4M2 23661615 IC50 = 7.8 nM T99840 CCX9Y5 23661672 IC50 = 5 nM T99840 CP93XI 23661699 IC50 = 2.4 nM T99840 CE5QD9 24180447 IC50 = 19600 nM T99840 C6FM9C 24180452 IC50 = 6.9 nM T99840 CB7ZC2 24180609 IC50 = 93 nM T99840 CK71ZR 24767800 IC50 = 2700 nM T99840 C8G7JD 24768566 IC50 = 96000 nM T99840 C3AM6Z 24779751 IC50 = 4.4 nM T99840 C03HRN 24864172 IC50 = 22 nM T99840 CE8DS6 24864173 IC50 = 220 nM T99840 CCX4P2 24864336 IC50 = 1.2 nM T99840 CK6E5Q 24864337 IC50 = 2 nM T99840 CVRN07 24864341 IC50 = 290 nM T99840 CG5CA4 24864523 IC50 = 1.6 nM T99840 C1V7WL 24864526 IC50 = 0.74 nM T99840 CIXE60 24864527 IC50 = 140 nM T99840 CDOV21 24864705 IC50 = 0.36 nM T99840 CK17JW 24864708 IC50 = 1.4 nM T99840 C8L0RO 24864709 IC50 = 2.1 nM T99840 CJ64HZ 24864711 IC50 = 0.17 nM T99840 CHG7C1 24864885 IC50 = 0.21 nM T99840 CREF30 24864886 IC50 = 0.28 nM T99840 CK2R6U 24865064 IC50 = 0.93 nM T99840 CJ1I9X 24865066 IC50 = 4.5 nM T99840 CGJ2Q4 24865068 IC50 = 2.6 nM T99840 CQ24JB 24865069 IC50 = 27 nM T99840 C1XP9G 24865249 IC50 = 0.52 nM T99840 CM17UV 24865251 IC50 = 1.1 nM T99840 CR8DV9 24865253 IC50 = 0.42 nM T99840 C26BIY 24865786 IC50 = 1.3 nM T99840 CN7GO5 24865789 IC50 = 2.4 nM T99840 C3HE0S 24865989 IC50 = 280 nM T99840 CSID98 24865993 IC50 = 85 nM T99840 C7I4VC 24866171 IC50 = 40 nM T99840 C48OQZ 24866173 IC50 = 0.46 nM T99840 CY0UC2 24866175 IC50 = 2.1 nM T99840 CZ1O3X 24866342 IC50 = 0.76 nM T99840 CE1FY8 24866343 IC50 = 5500 nM T99840 CP40OT 24866346 IC50 = 24 nM T99840 C8C5JG 24896257 IC50 = 5.6 nM T99840 C79GSB 24936138 IC50 = 0.32 nM T99840 C0B5LM 24936139 IC50 = 5.6 nM T99840 CKYX49 24963625 IC50 = 880 nM T99840 CU38IK 24964342 IC50 = 710 nM T99840 CQ7UB1 24964343 IC50 = 230 nM T99840 CXE6Q3 24964696 IC50 = 490 nM T99840 CWO1V4 25004449 IC50 = 840 nM T99840 CJR3M7 25014542 IC50 = 15000 nM T99840 CZ7G9O 25024968 IC50 = 28840 nM T99840 C5C7KU 25025157 IC50 > 50000 nM T99840 CG8WN5 25032613 IC50 = 0.27 nM T99840 C86CQY 25052759 IC50 = 214 nM T99840 CP7MH1 25106114 IC50 = 339 nM T99840 C98CGM 25106115 IC50 = 136 nM T99840 CLD7X0 25107258 IC50 = 898 nM T99840 C4NE6H 25107259 IC50 = 880 nM T99840 COT5G4 25107260 IC50 = 789 nM T99840 CL4XY0 25125138 IC50 = 2770 nM T99840 CIYA24 25125139 IC50 = 440 nM T99840 CH6Q5L 25125140 IC50 = 1440 nM T99840 C56EUJ 25138385 IC50 = 11 nM T99840 CW3OC1 25143875 IC50 = 58 nM T99840 C3DY8R 25144288 IC50 = 15 nM T99840 C2H4KJ 25145553 IC50 = 58 nM T99840 C3SOU5 25145846 IC50 = 75 nM T99840 CTF47W 25164607 IC50 = 1.3 nM T99840 CLW81T 25164608 IC50 = 7.4 nM T99840 CTB5M4 25164609 IC50 = 2 nM T99840 CQK4J3 25164810 IC50 = 6.4 nM T99840 CIJ2P5 25164811 IC50 = 6.8 nM T99840 CEKW51 25164812 IC50 = 5.5 nM T99840 C76DCT 25165012 IC50 = 25 nM T99840 C51XTP 25165014 IC50 = 0.9 nM T99840 C4ZJQ7 25165409 IC50 = 2.9 nM T99840 C3OIX5 25165410 IC50 = 1.4 nM T99840 CIXD52 25165995 IC50 = 63 nM T99840 C87EJY 25166594 IC50 = 5100 nM T99840 CVW64A 25166800 IC50 = 360 nM T99840 CSMD23 25186150 IC50 = 56 nM T99840 C52CEB 25186926 IC50 = 2 nM T99840 C2CTD9 25187263 IC50 = 135 nM T99840 CJL7I6 25225345 IC50 = 446 nM T99840 C82QUJ 25255222 IC50 = 144 nM T99840 CYOM53 25255427 IC50 = 94 nM T99840 C8TU1B 25255724 IC50 = 139 nM T99840 CD2GN0 25256437 IC50 = 322 nM T99840 CHP5E1 25256439 IC50 = 864 nM T99840 C4LMN1 25256522 IC50 = 955 nM T99840 C6J2PH 25256523 IC50 = 671 nM T99840 CO91CG 25263468 IC50 = 1 nM T99840 C4J1HV 25263469 IC50 = 0.65 nM T99840 C47ASX 25263470 IC50 = 0.51 nM T99840 CG4AI6 25263471 IC50 = 1.1 nM T99840 C83NHE 25263472 IC50 = 0.36 nM T99840 CKD1S7 25263473 IC50 = 1.9 nM T99840 CBY15W 25263474 IC50 = 35 nM T99840 CZ0TO9 25263475 IC50 = 0.82 nM T99840 CN65HK 25263476 IC50 = 0.25 nM T99840 C6Q5GS 25263477 IC50 = 0.66 nM T99840 C74ACU 25263478 IC50 = 0.15 nM T99840 C7RD5S 25263479 IC50 = 15 nM T99840 CP96SY 25263480 IC50 = 10 nM T99840 CW74XQ 25263481 IC50 = 2.1 nM T99840 CZ40XH 25263482 IC50 = 12 nM T99840 CT2MI1 25263483 IC50 = 15 nM T99840 CQL04P 25263484 IC50 = 12 nM T99840 CX3N1M 25263485 IC50 = 18 nM T99840 CRI45P 25263486 IC50 = 1.8 nM T99840 CC2FN6 25263487 IC50 = 0.93 nM T99840 CSKO45 25263488 IC50 = 4 nM T99840 CFH95Q 25263489 IC50 = 7.7 nM T99840 COIC78 25263490 IC50 = 0.06 nM T99840 C74LDY 25263491 IC50 = 0.06 nM T99840 C1WL7C 25263492 IC50 = 19 nM T99840 CIJU03 25263493 IC50 = 1.2 nM T99840 CF61JK 25263494 IC50 = 0.66 nM T99840 CP4TF9 25263495 IC50 = 0.41 nM T99840 CGO2Q4 25263496 IC50 = 0.48 nM T99840 CYG7A3 25263497 IC50 = 0.51 nM T99840 CZ2T1W 42632633 IC50 = 50.12 nM T99840 CZR8L4 42632635 IC50 = 63.1 nM T99840 C67ZYN 42632637 IC50 = 50.12 nM T99840 CS95DW 42632653 IC50 = 63.1 nM T99840 CM8OV5 42632655 IC50 = 199.53 nM T99840 CSGK56 42632682 IC50 = 316.23 nM T99840 CXD8G0 42632750 IC50 = 199.53 nM T99840 C5QE0V 42632752 IC50 = 630.96 nM T99840 C05NRU 42632754 IC50 = 158.49 nM T99840 CEVN24 42632772 IC50 = 316.23 nM T99840 CT8L3J 42632842 IC50 = 125.89 nM T99840 C6NZ5A 42632900 IC50 = 125.89 nM T99840 C87POD 42633502 IC50 = 116 nM T99840 CAX43F 42633863 IC50 = 509 nM T99840 C0S8GC 42638432 IC50 = 500 nM T99840 CZS65J 42638433 IC50 = 1200 nM T99840 CH3MY1 42639933 IC50 = 260 nM T99840 CVY8H2 42640092 IC50 = 460 nM T99840 CU68PM 42640420 IC50 = 170 nM T99840 CRGV67 42640423 IC50 = 540 nM T99840 CT0OU1 42640598 IC50 = 2780 nM T99840 C2MY8X 42647277 IC50 = 44 nM T99840 CX3L0P 44139437 IC50 = 8.81 nM T99840 C3ZGR9 44157625 IC50 = 0.46 nM T99840 CA9FN6 44193857 IC50 = 209 nM T99840 CE5A9Z 44193858 IC50 = 133 nM T99840 CFEX37 44193859 IC50 = 244 nM T99840 CBC3W9 44193860 IC50 = 252 nM T99840 C19RXP 44193960 IC50 = 212 nM T99840 CEM1J3 44193962 IC50 = 127 nM T99840 CU06VM 44193963 IC50 = 651 nM T99840 CE1PW4 44194155 IC50 = 319 nM T99840 CBS1D6 44195184 IC50 = 133 nM T99840 C5T3FW 44195186 IC50 = 123 nM T99840 CV6WM1 44241633 IC50 = 154 nM T99840 C3SFT9 44272269 IC50 = 5000 nM T99840 CA4F7H 44272270 IC50 = 3400 nM T99840 C7EQ2R 44272404 IC50 = 400 nM T99840 CL15MO 44272482 IC50 = 15000 nM T99840 CL4J3Z 44272483 IC50 = 180 nM T99840 C6L1IY 44272484 IC50 = 400 nM T99840 CS67FV 44272499 IC50 = 1500 nM T99840 CQHE15 44272500 IC50 = 1600 nM T99840 CK5EV7 44272502 IC50 = 550 nM T99840 C3HB6A 44272553 IC50 = 580 nM T99840 CP3NY6 44272576 IC50 = 620 nM T99840 C81DBR 44272577 IC50 = 15000 nM T99840 C0ME2L 44272578 IC50 = 450 nM T99840 CQYN68 44272595 IC50 = 300 nM T99840 C48XAS 44272596 IC50 = 17000 nM T99840 C9W6EG 44272620 IC50 > 25000 nM T99840 C8DG3U 44272639 IC50 > 25000 nM T99840 CTJ28F 44272794 IC50 > 25000 nM T99840 C6I7FY 44272815 IC50 = 3300 nM T99840 CA5C6N 44272822 IC50 = 600 nM T99840 C1ARU0 44272823 IC50 = 900 nM T99840 C79FBO 44272863 IC50 = 920 nM T99840 CL0PB6 44272874 IC50 = 1800 nM T99840 CL08UE 44299780 IC50 = 1200 nM T99840 CIMP62 44299785 IC50 = 240 nM T99840 CTP4K5 44299806 IC50 = 150 nM T99840 CFDX15 44299807 IC50 = 800 nM T99840 CO58LY 44299816 IC50 = 1100 nM T99840 C72ICU 44299831 IC50 = 6 nM T99840 CD4K9L 44299838 IC50 = 480 nM T99840 C4JC6H 44299839 IC50 = 4.7 nM T99840 CB9W1F 44299856 IC50 > 2500 nM T99840 CI8H6V 44299857 IC50 = 454 nM T99840 CSBE57 44299884 IC50 = 1000 nM T99840 CD7K6U 44299900 IC50 > 2500 nM T99840 C4IB5Y 44299922 IC50 = 20 nM T99840 CQIZ85 44299941 IC50 = 408 nM T99840 CCZ5H7 44299970 IC50 = 3200 nM T99840 C8AJ3U 44299981 IC50 = 240 nM T99840 CEBH91 44299982 IC50 > 2600 nM T99840 CO26SB 44299986 IC50 = 160 nM T99840 C34TQN 44299987 IC50 = 71 nM T99840 C72LXP 44300008 IC50 = 1700 nM T99840 C9JUG3 44300019 IC50 > 2500 nM T99840 CHV7K8 44300020 IC50 = 66 nM T99840 C06ZXT 44300027 IC50 > 2500 nM T99840 C45QVN 44300045 IC50 = 300 nM T99840 CD6VT9 44300046 IC50 = 32 nM T99840 CH3BD1 44300054 IC50 > 2500 nM T99840 C37NVU 44300062 IC50 = 2400 nM T99840 C9B4TQ 44300116 IC50 = 280 nM T99840 C3G7CU 44300117 IC50 = 900 nM T99840 CDUB40 44300118 IC50 = 800 nM T99840 C1MW5E 44300137 IC50 = 50 nM T99840 C6IAU4 44300141 IC50 = 102 nM T99840 C43QHF 44300156 IC50 = 55 nM T99840 C6OT5P 44300185 IC50 = 52 nM T99840 CZX60N 44300200 IC50 = 36 nM T99840 C4F9SV 44300201 IC50 > 2500 nM T99840 CU82ZK 44300204 IC50 > 2500 nM T99840 CW3M8K 44300206 IC50 > 2500 nM T99840 C1C0FH 44300213 IC50 > 2500 nM T99840 CM5Y2D 44300220 IC50 > 2500 nM T99840 C04MOF 44300225 IC50 = 2000 nM T99840 CEFA26 44300242 IC50 = 1 nM T99840 CFJ3S7 44300372 IC50 > 2500 nM T99840 CPKU38 44300560 IC50 = 300 nM T99840 CKE03P 44300566 IC50 = 13 nM T99840 CDJ1K4 44300571 IC50 = 130 nM T99840 CZ29RH 44300582 IC50 = 39 nM T99840 CMOE73 44300584 IC50 = 17 nM T99840 C8CT2N 44344777 IC50 = 140 nM T99840 CAK7D0 44344792 IC50 = 57 nM T99840 CA6G8L 44344798 IC50 = 720 nM T99840 CMV09U 44344902 IC50 > 2500 nM T99840 CVH04W 44344916 IC50 = 5 nM T99840 C3S7ZH 44344917 IC50 = 14 nM T99840 C4KUV7 44344918 IC50 = 38 nM T99840 CPZ1M7 44344923 IC50 = 86 nM T99840 CM4FQ2 44344936 IC50 > 2500 nM T99840 C4L6GK 44344979 IC50 = 47 nM T99840 CG3TN7 44344993 IC50 = 1500 nM T99840 C4YU7O 44345078 IC50 = 4 nM T99840 CTD02F 44345083 IC50 = 37 nM T99840 CJ0R9G 44345100 IC50 = 190 nM T99840 CBQ50F 44345133 IC50 = 150 nM T99840 CHZ46Y 44345144 IC50 > 2500 nM T99840 CXPR42 44345153 IC50 > 2500 nM T99840 CI7B2O 44345154 IC50 > 2500 nM T99840 C2OE7B 44354160 IC50 = 1884 nM T99840 C93ODM 44354173 IC50 = 100.6 nM T99840 C72GNU 44354186 IC50 = 4.7 nM T99840 C4IL1K 44354199 IC50 = 2.2 nM T99840 C0ICU7 44354337 IC50 = 5.5 nM T99840 C93ZCV 44354338 IC50 = 28 nM T99840 CJPT35 44354363 IC50 = 12.7 nM T99840 C6FDY5 44354364 IC50 = 1.8 nM T99840 CSFK05 44354431 IC50 = 0.49 nM T99840 CIF9Q4 44354432 IC50 = 0.9 nM T99840 CMG1C8 44354433 IC50 = 3.7 nM T99840 CSM8K2 44354444 IC50 = 13.2 nM T99840 CGJU57 44354445 IC50 = 1.2 nM T99840 CQY1M8 44354459 IC50 = 1.8 nM T99840 C0VL9I 44354463 IC50 = 3.6 nM T99840 CD02RP 44354512 IC50 = 0.3 nM T99840 CK2I9B 44386459 IC50 = 400 nM T99840 C0K1RP 44386460 IC50 = 390 nM T99840 C1DIV7 44386461 IC50 = 18000 nM T99840 C5Q8HR 44386506 IC50 = 230 nM T99840 C97HRQ 44386664 IC50 = 8000 nM T99840 CB7C4E 44386766 IC50 = 20000 nM T99840 CE6Y3A 44386767 IC50 = 250 nM T99840 CQ4LM3 44386768 IC50 = 150 nM T99840 CC0MF8 44386780 IC50 = 22000 nM T99840 CZ51MR 44386781 IC50 = 400 nM T99840 C4TY6U 44386828 IC50 = 140 nM T99840 CU9TH3 44386902 IC50 = 500 nM T99840 C0NRO6 44387006 IC50 = 670 nM T99840 CBHG04 44387127 IC50 = 530 nM T99840 C67JZV 44387228 IC50 = 540 nM T99840 C7J2SN 44388746 IC50 = 152 nM T99840 CLY7C6 44388755 IC50 = 623 nM T99840 C1LJ6O 44388757 IC50 = 39 nM T99840 CE85NT 44388765 IC50 = 335 nM T99840 CQL81R 44388767 IC50 = 21 nM T99840 C8RJW0 44388774 IC50 = 15 nM T99840 C4F3XD 44388775 IC50 = 209 nM T99840 C4OS5H 44388781 IC50 = 5 nM T99840 CSD0H2 44391778 IC50 > 1000 nM T99840 CCTX25 44391779 IC50 = 62 nM T99840 CMD12V 44391780 IC50 = 29 nM T99840 CW1M4K 44391785 IC50 > 1000 nM T99840 C56HFN 44391787 IC50 = 16 nM T99840 CH0YT8 44391790 IC50 > 1000 nM T99840 CGZ06W 44391795 IC50 = 75 nM T99840 CX1Z5Y 44391797 IC50 > 1000 nM T99840 CEJ6X3 44391801 IC50 = 6 nM T99840 C9WSN6 44391803 IC50 > 1000 nM T99840 CPM3E0 44391804 IC50 = 721 nM T99840 CKD81U 44391806 IC50 = 34 nM T99840 C17PFC 44391809 IC50 = 239 nM T99840 CJT3D5 44391810 IC50 = 12 nM T99840 C1VP5T 44391812 IC50 = 146 nM T99840 C9N8MZ 44391813 IC50 = 412 nM T99840 CA5H3N 44391817 IC50 = 535 nM T99840 CR3D5J 44391818 IC50 = 7 nM T99840 C7HL9Y 44391819 IC50 = 610 nM T99840 C6ZJW2 44391822 IC50 = 324 nM T99840 CA59PK 44391823 IC50 > 1000 nM T99840 CQ23WT 44391825 IC50 = 175 nM T99840 CMQ25A 44391827 IC50 = 129 nM T99840 C3O7NC 44391829 IC50 = 153 nM T99840 C7KX2F 44391831 IC50 > 1000 nM T99840 CY45WQ 44391832 IC50 = 41 nM T99840 CX68DF 44391834 IC50 = 490 nM T99840 C9KPT6 44391836 IC50 > 1000 nM T99840 C6OD3B 44391837 IC50 = 269 nM T99840 CC0N5Q 44391839 IC50 > 1000 nM T99840 CVM40E 44391840 IC50 = 74 nM T99840 CP6A0L 44391845 IC50 = 69 nM T99840 COMI50 44391846 IC50 > 1000 nM T99840 CL8IU7 44391850 IC50 > 1000 nM T99840 C2GL0H 44391851 IC50 = 467 nM T99840 CM5G8L 44391852 IC50 = 23 nM T99840 CLT4I7 44391857 IC50 > 1000 nM T99840 CVOC09 44391862 IC50 = 3490 nM T99840 C0U6SQ 44391880 IC50 = 73 nM T99840 CR95TU 44391894 IC50 = 227 nM T99840 CGC76F 44391900 IC50 = 5 nM T99840 CT9N4H 44391911 IC50 = 226 nM T99840 CS19FK 44396232 IC50 = 25 nM T99840 C2ZVO0 44400673 IC50 = 12 nM T99840 C1K2IX 44400710 IC50 = 104 nM T99840 CUSQ68 44400771 IC50 = 170 nM T99840 C7Z5DM 44400772 IC50 = 27 nM T99840 C10QIO 44400790 IC50 = 55 nM T99840 C4V0IG 44400842 IC50 = 253 nM T99840 CTFY61 44400878 IC50 = 98 nM T99840 C8SO5T 44400879 IC50 = 1900 nM T99840 CPVJ60 44400904 IC50 = 2472 nM T99840 C4DBM3 44400933 IC50 = 249 nM T99840 C75GIF 44403333 IC50 = 62 nM T99840 C1UJK7 44403341 IC50 = 132 nM T99840 CGMY50 44403342 IC50 = 1 nM T99840 C3Y5PS 44403401 IC50 = 394 nM T99840 C89GRJ 44403409 IC50 = 766 nM T99840 CTC17R 44403410 IC50 = 134 nM T99840 C9ZSM3 44403413 IC50 = 429 nM T99840 CDA16M 44403414 IC50 = 138 nM T99840 C9Z2TM 44403415 IC50 = 122 nM T99840 CJSH92 44403418 IC50 = 17 nM T99840 C0YSJ9 44403419 IC50 = 19 nM T99840 C7TYW4 44403423 IC50 = 2 nM T99840 CY61LD 44403424 IC50 = 3.4 nM T99840 COVL82 44403428 IC50 = 250 nM T99840 CMZ25N 44403431 IC50 = 18 nM T99840 C7XJ8T 44403432 IC50 = 21 nM T99840 CK09NJ 44403434 IC50 = 4 nM T99840 CF7LQ4 44411586 IC50 = 1.39 nM T99840 CJA03K 44411650 IC50 = 0.24 nM T99840 CXG72Q 44411651 IC50 = 0.76 nM T99840 CPTX52 44411690 IC50 = 0.04 nM T99840 C2OS3K 44411691 IC50 = 0.08 nM T99840 CP9T4I 44411692 IC50 = 0.06 nM T99840 CY9BW4 44412059 IC50 = 0.4 nM T99840 CCD8N4 44412061 IC50 = 1.17 nM T99840 CH0O5Z 44412062 IC50 = 0.41 nM T99840 C79ZOD 44412080 IC50 = 0.19 nM T99840 C30DSF 44412081 IC50 = 0.9 nM T99840 C6HDY0 44412083 IC50 = 0.26 nM T99840 CMNE06 44412297 IC50 = 6.18 nM T99840 C85GSO 44413510 IC50 > 100000 nM T99840 CDM4F2 44413568 IC50 > 100000 nM T99840 C13BKF 44413569 IC50 = 500 nM T99840 C58TNH 44413653 IC50 = 85 nM T99840 C26HYC 44413654 IC50 = 8 nM T99840 CJ4U8X 44413659 IC50 > 100000 nM T99840 CJXW54 44413660 IC50 = 4600 nM T99840 C0K8UY 44413669 IC50 = 112 nM T99840 C4X5BG 44413670 IC50 = 24 nM T99840 CFU14K 44413689 IC50 = 380 nM T99840 CZ3B4H 44413690 IC50 = 10 nM T99840 CG5N4R 44413701 IC50 = 210 nM T99840 CB52ER 44413711 IC50 = 44 nM T99840 CDG6W4 44413753 IC50 = 1628 nM T99840 C4TZ7D 44413785 IC50 = 7200 nM T99840 CL7Y8W 44413786 IC50 = 5900 nM T99840 C8HUB4 44413791 IC50 = 376 nM T99840 CM6D4R 44413792 IC50 = 77 nM T99840 C21BHJ 44413797 IC50 > 100000 nM T99840 CAV8Z0 44413798 IC50 = 26000 nM T99840 C87MVI 44413804 IC50 = 55 nM T99840 CW8CK0 44413805 IC50 = 10 nM T99840 CQ4NY3 44413810 IC50 > 100000 nM T99840 CJP10D 44413812 IC50 > 100000 nM T99840 CTM24D 44413821 IC50 > 100000 nM T99840 C1O3DB 44413822 IC50 > 100000 nM T99840 C0PZ4N 44414662 IC50 = 1000 nM T99840 C60SKV 44414672 IC50 = 1100 nM T99840 C6GV4A 44414676 IC50 = 130 nM T99840 CN0S8T 44414677 IC50 = 17000 nM T99840 CW73JT 44414685 IC50 = 490 nM T99840 C4JD8U 44414686 IC50 = 10 nM T99840 C3U0HO 44414698 IC50 = 530 nM T99840 C7Z2DP 44414744 IC50 = 3200 nM T99840 CEVF60 44414745 IC50 = 10 nM T99840 C6PA2W 44414746 IC50 = 20 nM T99840 C96UKI 44414773 IC50 = 4400 nM T99840 CJ3H8L 44414774 IC50 = 1300 nM T99840 CX15LW 44414778 IC50 = 6.1 nM T99840 CF3E7Y 44414797 IC50 = 470 nM T99840 CNI3J4 44414807 IC50 = 530 nM T99840 C8LKZ2 44414808 IC50 = 350 nM T99840 CG4MU6 44414826 IC50 = 400 nM T99840 CKHW96 44414838 IC50 = 1900 nM T99840 CM68NQ 44414839 IC50 = 690 nM T99840 C5HG7K 44414857 IC50 = 1200 nM T99840 CLSE91 44414858 IC50 = 3000 nM T99840 C1AGV6 44421238 IC50 = 200 nM T99840 CCKQ89 44421239 IC50 = 7000 nM T99840 C7BA5U 44421240 IC50 = 2000 nM T99840 CPY82H 44421241 IC50 = 3000 nM T99840 C9VH0I 44421242 IC50 = 3000 nM T99840 CO9XG3 44421243 IC50 = 2000 nM T99840 CF64CH 44421244 IC50 = 24000 nM T99840 C2ACK0 44421245 IC50 = 12000 nM T99840 C6PXS2 44421246 IC50 = 3000 nM T99840 CG7V9P 44421321 IC50 = 900 nM T99840 CADE57 44421322 IC50 = 2000 nM T99840 CL13AF 44421323 IC50 = 6000 nM T99840 C6G0XP 44421334 IC50 = 5000 nM T99840 C9R0TM 44421335 IC50 = 600 nM T99840 CCJB73 44429704 IC50 = 2500 nM T99840 CM6GO3 44429705 IC50 = 680 nM T99840 C46SOY 44429706 IC50 = 270 nM T99840 CHR0P6 44429707 IC50 = 15420 nM T99840 C1I2WC 44429708 IC50 = 219 nM T99840 C3MLB9 44429709 IC50 = 159 nM T99840 CDOV06 44429710 IC50 = 34 nM T99840 C73NZY 44429711 IC50 = 12300 nM T99840 CL23CT 44429712 IC50 = 4770 nM T99840 CNEI43 44429713 IC50 = 71 nM T99840 CUK8Q2 44429715 IC50 = 37 nM T99840 C2CB3A 44429716 IC50 = 38 nM T99840 C73HBA 44429717 IC50 = 26 nM T99840 C9I5KO 44429718 IC50 = 13 nM T99840 C0XP3E 44429723 IC50 = 28 nM T99840 C83NCX 44429724 IC50 = 10 nM T99840 CE8U1T 44429726 IC50 = 36 nM T99840 CUQ1P7 44429727 IC50 = 7 nM T99840 CHZY93 44429728 IC50 = 4 nM T99840 CQ5WV3 44429729 IC50 = 26 nM T99840 C71IMA 44429730 IC50 = 8 nM T99840 C9ZGA2 44432541 Ki = 1000 nM T99840 CW2GR3 44432543 Ki = 227 nM T99840 CFWE67 44432548 Ki = 15 nM T99840 CS4BO0 44432549 Ki = 11 nM T99840 CDE85L 44432550 Ki = 3.5 nM T99840 C4JO5H 44432551 Ki = 1.2 nM T99840 C6ZF0L 44432552 Ki = 1.4 nM T99840 CGH6N0 44432554 Ki = 6.2 nM T99840 C4H9BC 44432556 Ki = 2 nM T99840 CC5L7X 44432557 Ki = 3 nM T99840 CK52RJ 44432568 IC50 = 19 nM T99840 CV3FY9 44432569 Ki = 36 nM T99840 C6G2BA 44432572 Ki = 9.9 nM T99840 C36YRT 44432575 Ki = 13.5 nM T99840 CY6CL0 44432578 Ki = 4.9 nM T99840 CM3DJ5 44432579 Ki = 4 nM T99840 C6KUW0 44432584 Ki = 2.2 nM T99840 CE1W6U 44432588 Ki = 1.3 nM T99840 CP24YK 44432590 Ki = 1.1 nM T99840 C89PTY 44432592 Ki = 3.9 nM T99840 C67PIK 44432596 Ki = 2.1 nM T99840 CE8US0 44432598 Ki = 0.9 nM T99840 CMA4O9 44432601 Ki = 22 nM T99840 C4DR0K 44432604 Ki = 3.1 nM T99840 C3XBU0 44432607 Ki = 111 nM T99840 CD0ET2 44432735 IC50 = 850 nM T99840 CH73FO 44432736 IC50 = 1100 nM T99840 CJY57U 44432737 IC50 = 750 nM T99840 C2SYG0 44432738 IC50 = 1300 nM T99840 C8FGR3 44432739 IC50 = 400 nM T99840 CDW4U1 44432740 IC50 = 700 nM T99840 C4I3RA 44432741 IC50 = 2000 nM T99840 C92DVC 44432742 IC50 = 920 nM T99840 CUC3O6 44432743 IC50 = 1000 nM T99840 CQ6G1T 44432744 IC50 = 350 nM T99840 CM17EH 44432745 IC50 = 190 nM T99840 C4FC1D 44432746 IC50 = 1000 nM T99840 C7QP9I 44432747 IC50 = 1200 nM T99840 CIJ31A 44432748 IC50 = 360 nM T99840 CU4LA7 44432749 IC50 = 720 nM T99840 CR78GI 44432750 IC50 = 1200 nM T99840 C5MR7Y 44432751 IC50 = 66 nM T99840 CIR93O 44432752 IC50 = 56 nM T99840 C2SUF9 44432753 IC50 = 19 nM T99840 C7GUX6 44432754 IC50 = 72 nM T99840 CLP08T 44432755 IC50 = 180 nM T99840 CSM3Y2 44432757 IC50 = 1300 nM T99840 CY2OV0 44432758 IC50 = 240 nM T99840 C6E1LT 44432759 IC50 = 560 nM T99840 CZKR96 44432760 IC50 > 25000 nM T99840 CFL9M6 44432780 IC50 = 13 nM T99840 C39CUV 44432782 IC50 = 140 nM T99840 CTZ64S 44432784 IC50 = 23 nM T99840 CQ1UV3 44432785 IC50 = 25 nM T99840 CT2JH3 44432787 IC50 = 7 nM T99840 CNC96Y 44432789 IC50 = 49 nM T99840 CK70ES 44432792 IC50 = 12 nM T99840 CNFB80 44432793 IC50 = 14 nM T99840 C06KEF 44432796 IC50 = 33 nM T99840 C68JBI 44432797 IC50 = 22 nM T99840 CNQ2X3 44432799 IC50 = 41 nM T99840 C4DHY0 44432800 IC50 = 100 nM T99840 CG7MS6 44432801 IC50 = 140 nM T99840 C80GXR 44432802 IC50 = 1300 nM T99840 CK5IO0 44432804 IC50 = 100 nM T99840 CN21WE 44432805 IC50 = 3700 nM T99840 CTZD96 44432807 IC50 = 24 nM T99840 CV4GI8 44432808 IC50 = 14 nM T99840 C1Z9UG 44432809 IC50 = 4 nM T99840 CV9AI5 44432810 IC50 = 5 nM T99840 C7PEV0 44433881 IC50 = 1500 nM T99840 C7JQW3 44433888 IC50 = 3.1 nM T99840 CZ8K2R 44433889 IC50 = 580 nM T99840 CNKB48 44433891 IC50 = 1.6 nM T99840 CCGZ80 44433893 IC50 = 7.1 nM T99840 CZ8G4V 44433896 IC50 = 5.3 nM T99840 CH0PB4 44433897 IC50 = 6.3 nM T99840 CE1BP2 44433898 IC50 = 12 nM T99840 C7TD8Q 44433899 IC50 = 22 nM T99840 CP19WA 44433901 IC50 = 20 nM T99840 CC76FQ 44433923 IC50 = 0.002 nM T99840 C7HSE9 44433930 IC50 = 1.7 nM T99840 C4Q2MH 44435366 IC50 = 27 nM T99840 CX51JK 44435367 IC50 = 12 nM T99840 C1SCL8 44435394 IC50 = 11.6 nM T99840 CVF83U 44435448 IC50 = 0.3 nM T99840 CO16ME 44435449 IC50 = 0.3 nM T99840 CT3NY9 44435450 IC50 = 7.49 nM T99840 C4CBZ6 44435451 IC50 = 0.05 nM T99840 C2TX3S 44435452 IC50 = 0.14 nM T99840 C4PM7B 44435453 IC50 = 30 nM T99840 C3UA0C 44435454 IC50 = 81.5 nM T99840 C54DVE 44435455 IC50 = 0.22 nM T99840 CW1O9L 44435456 IC50 = 0.22 nM T99840 CJO6U3 44435457 IC50 = 0.43 nM T99840 COB67F 44435458 IC50 = 0.11 nM T99840 CK84MV 44435459 IC50 = 1.14 nM T99840 C92MHT 44435460 IC50 = 50.5 nM T99840 C6PHM1 44435462 IC50 = 63.2 nM T99840 CWZ10L 44435463 IC50 = 42 nM T99840 C0QIS7 44435464 IC50 = 4.5 nM T99840 CY2V0F 44435465 IC50 = 10.1 nM T99840 C94BOF 44435466 IC50 = 29.8 nM T99840 C97KQX 44435467 IC50 = 2 nM T99840 C9U6ZV 44435468 IC50 = 7.1 nM T99840 CI4R2T 44435469 IC50 = 4.2 nM T99840 C3R4SW 44435470 IC50 = 3.1 nM T99840 CZ4L1H 44435471 IC50 = 134 nM T99840 CWF51G 44435472 IC50 = 2.6 nM T99840 CO17MG 44435473 IC50 = 5 nM T99840 CMVY01 44435474 IC50 = 2.7 nM T99840 CO7PI4 44435475 IC50 = 5.9 nM T99840 CBG0P2 44435476 IC50 = 28.3 nM T99840 C7VGP3 44435477 IC50 = 1.4 nM T99840 CKJV32 44435478 IC50 = 4 nM T99840 COHJ47 44435479 IC50 = 30 nM T99840 C0YU6V 44435480 IC50 = 10 nM T99840 C4KC1T 44435481 IC50 = 30 nM T99840 CFWA70 44435482 IC50 = 2.4 nM T99840 CD1H4G 44435483 IC50 = 26.1 nM T99840 C8DZ0C 44435484 IC50 = 30 nM T99840 CK95FN 44435485 IC50 = 2.2 nM T99840 CNXB96 44435486 IC50 = 1 nM T99840 C61BSW 44435487 IC50 < 34.6 nM T99840 CFLH45 44435488 IC50 = 64.8 nM T99840 C3VC7X 44435489 IC50 = 2.8 nM T99840 C8J2WB 44435490 IC50 = 141 nM T99840 CA9F6R 44435491 IC50 = 0.3 nM T99840 C4A5HJ 44435492 IC50 = 141 nM T99840 CCID56 44435493 IC50 = 12.9 nM T99840 CIO39Q 44435494 IC50 = 27.7 nM T99840 CX29JY 44435495 IC50 = 20.1 nM T99840 CXTH68 44435496 IC50 = 37.3 nM T99840 C32ZBN 44435497 IC50 = 16.8 nM T99840 C8ZU7E 44435530 IC50 = 13.6 nM T99840 CT6DY8 44438312 IC50 = 7.7 nM T99840 CJW0F5 44438313 IC50 = 26.8 nM T99840 C9YL5C 44438316 IC50 = 74.8 nM T99840 C4Q9NI 44438319 IC50 = 110 nM T99840 C6W2IH 44438321 IC50 = 152.5 nM T99840 C5GQ4C 44438322 IC50 = 164.5 nM T99840 CTYV56 44438323 IC50 = 0.7 nM T99840 C6Z9MA 44438324 IC50 = 5.3 nM T99840 CMJ73E 44438325 IC50 = 4.2 nM T99840 CU13SQ 44438327 IC50 = 7.9 nM T99840 C9B1UA 44438328 IC50 = 6.1 nM T99840 C97WJB 44438331 IC50 = 8.5 nM T99840 CET92A 44438332 IC50 = 15.4 nM T99840 CCQ4L2 44438334 IC50 = 3.7 nM T99840 C03BAR 44438335 IC50 = 4.5 nM T99840 C5S0ZB 44438337 IC50 = 5.5 nM T99840 CJW68H 44438338 IC50 = 9.7 nM T99840 C4A1IW 44438339 IC50 = 5.2 nM T99840 CR0WN3 44438340 IC50 = 3.6 nM T99840 CUTO72 44438341 IC50 = 120.4 nM T99840 C5PTA0 44438342 IC50 = 1.9 nM T99840 C2CYK4 44438343 IC50 = 2.1 nM T99840 C6AR1L 44438344 IC50 = 0.9 nM T99840 CH1A9C 44438345 IC50 = 0.3 nM T99840 CI9Z5D 44438347 IC50 = 16.8 nM T99840 CY4JS2 44438348 IC50 = 2.7 nM T99840 CQ1D4N 44438349 IC50 = 1.1 nM T99840 C5V0SU 44438350 IC50 = 2.4 nM T99840 CL5R1O 44438351 IC50 = 3.5 nM T99840 CVL65S 44438352 IC50 = 16.8 nM T99840 C7EV9J 44438385 IC50 = 172 nM T99840 C4QGK6 44438388 IC50 = 253 nM T99840 C5R0TJ 44438390 IC50 = 580 nM T99840 C7F6CI 44438393 IC50 = 440 nM T99840 CX8PM9 44438400 IC50 = 680 nM T99840 C1V4HC 44438402 IC50 = 629 nM T99840 CGAF37 44438404 IC50 = 290 nM T99840 CX0V5I 44438413 IC50 = 255 nM T99840 CW8R1G 44438417 IC50 = 219 nM T99840 CV98FE 44438419 IC50 = 217 nM T99840 C20UWR 44438421 IC50 > 1000 nM T99840 CTS16G 44438436 IC50 = 4.4 nM T99840 CFH2R8 44438651 IC50 = 13000 nM T99840 CLEM85 44438652 IC50 > 40000 nM T99840 C0JO3P 44438653 IC50 = 24000 nM T99840 C85LSF 44438654 IC50 = 38000 nM T99840 C0SWQ8 44438655 IC50 = 37000 nM T99840 CDHQ05 44438656 IC50 = 32000 nM T99840 CNQ7O0 44438657 IC50 = 13000 nM T99840 C5OS0L 44438658 IC50 > 40000 nM T99840 CCK6H4 44438659 IC50 = 16000 nM T99840 C3TEI7 44438660 IC50 = 19000 nM T99840 C73OXN 44438661 IC50 = 17000 nM T99840 CITL79 44438662 IC50 = 11000 nM T99840 CG9C3D 44440636 IC50 = 9 nM T99840 C7HY4S 44440637 IC50 = 6 nM T99840 CIPS34 44440638 IC50 = 8 nM T99840 C1RZ7M 44440639 IC50 = 59 nM T99840 C3XE9I 44440640 IC50 = 10 nM T99840 CN7H4Z 44440641 IC50 = 162 nM T99840 C7L8UV 44440642 IC50 = 43 nM T99840 CE7K6W 44440643 IC50 = 269 nM T99840 C1S3AI 44440644 IC50 = 3 nM T99840 CF1H9O 44440649 IC50 = 1 nM T99840 CJ5BS7 44440650 IC50 = 24 nM T99840 CH8P2F 44440651 IC50 = 1 nM T99840 C7WJL5 44440652 IC50 = 4 nM T99840 CK98ME 44440653 IC50 = 1.3 nM T99840 CN06BY 44440654 IC50 = 0.2 nM T99840 CSC65N 44440655 IC50 = 2 nM T99840 CY29QH 44440658 IC50 = 0.5 nM T99840 CV5T4N 44440666 IC50 = 2 nM T99840 CV3OC2 44440667 IC50 = 14 nM T99840 C7Z3TC 44440668 IC50 = 22 nM T99840 CRL40U 44440669 IC50 = 1.9 nM T99840 C29GPX 44440670 IC50 = 14 nM T99840 CTYP45 44440671 IC50 = 56 nM T99840 C9G1NJ 44440672 IC50 = 0.4 nM T99840 C86GRL 44440673 IC50 = 10 nM T99840 C0EM2O 44440674 IC50 = 750 nM T99840 CV6MS8 44441997 IC50 = 5.2 nM T99840 CDA0K3 44441998 IC50 = 18.5 nM T99840 C6VF9N 44441999 IC50 = 783 nM T99840 C5KPT0 44442000 IC50 > 1000 nM T99840 CSXU96 44442006 IC50 = 28.4 nM T99840 CF2NQ0 44442007 IC50 = 71.1 nM T99840 CX5V1C 44442008 IC50 = 103.5 nM T99840 C41NKY 44442009 IC50 > 1000 nM T99840 CH97AI 44442010 IC50 > 1000 nM T99840 C31THS 44442011 IC50 = 154.5 nM T99840 CPFY31 44442012 IC50 = 310.1 nM T99840 CWTI80 44442013 IC50 = 48.8 nM T99840 C4NST7 44442014 IC50 = 2.4 nM T99840 C3YR2W 44442017 IC50 = 8.1 nM T99840 C65KFB 44443276 EC50 = 10600 nM T99840 CFE6Y0 44443278 EC50 = 6200 nM T99840 CQLY72 44443990 IC50 = 3400 nM T99840 CI53PU 44443991 IC50 = 13 nM T99840 CB3O4E 44443992 IC50 = 3200 nM T99840 C7PEB3 44443993 IC50 = 9.7 nM T99840 CX96US 44443994 IC50 = 57 nM T99840 CU0A7X 44443995 IC50 = 9 nM T99840 CA2U1Z 44443997 IC50 = 830 nM T99840 CTX10R 44443998 IC50 = 7700 nM T99840 CL8VK6 44443999 IC50 = 180 nM T99840 C4V5PO 44444004 IC50 = 25 nM T99840 C7O1LX 44444015 IC50 = 21 nM T99840 CJD64U 44444017 IC50 = 65 nM T99840 CM95NK 44444020 IC50 = 13 nM T99840 C7ABX0 44444022 IC50 = 76 nM T99840 CKXE20 44444023 IC50 = 18 nM T99840 CXYJ51 44444048 IC50 = 45 nM T99840 CFAU69 44444049 IC50 = 33 nM T99840 CL18UT 44444050 IC50 = 12 nM T99840 CK2B9V 44444051 IC50 = 25 nM T99840 C3HGR6 44444054 IC50 = 41 nM T99840 C2UD9K 44444056 IC50 = 15 nM T99840 C63MJP 44444058 IC50 = 93 nM T99840 CED08T 44444059 IC50 = 29 nM T99840 CR43VX 44444063 IC50 = 64 nM T99840 C9BG8M 44444064 IC50 = 60 nM T99840 CC0Q9I 44444066 IC50 = 820 nM T99840 CM4FU3 44444067 IC50 = 660 nM T99840 CHTL58 44444068 IC50 = 130 nM T99840 CMXC12 44444069 IC50 = 550 nM T99840 CI8O7E 44444071 IC50 = 130 nM T99840 C49PGO 44444072 IC50 = 67 nM T99840 CLOY45 44444073 IC50 = 460 nM T99840 CL1HR0 44444074 IC50 = 120 nM T99840 C42NRC 44444075 IC50 = 340 nM T99840 CNI37J 44444077 IC50 = 27 nM T99840 C4CKQ7 44444078 IC50 = 690 nM T99840 C1YF2B 44444079 IC50 = 4500 nM T99840 C0YK9T 44444080 IC50 = 1400 nM T99840 C1DQN8 44444081 IC50 = 620 nM T99840 CDN8F5 44444082 IC50 = 110 nM T99840 CVG61I 44444083 IC50 = 85 nM T99840 CLP4E8 44444085 IC50 = 1100 nM T99840 CZ3O5X 44444087 IC50 = 67 nM T99840 C4J0ZO 44444088 IC50 = 470 nM T99840 CP0G8B 44444089 IC50 = 1000 nM T99840 CXD61J 44444090 IC50 = 330 nM T99840 C8TI3U 44444091 IC50 = 180 nM T99840 C7MTH4 44444092 IC50 = 150 nM T99840 CC2P1R 44444093 IC50 = 3900 nM T99840 C6CSF4 44444095 IC50 = 250 nM T99840 C1L2XV 44446139 IC50 = 5.1 nM T99840 CO57IE 44446141 IC50 = 7.3 nM T99840 CVOK90 44446142 IC50 = 13 nM T99840 C5T1SX 44446144 IC50 = 8.1 nM T99840 C0AEN8 44446145 IC50 = 6.9 nM T99840 CNGW15 44446147 IC50 = 14 nM T99840 CB52UA 44446149 IC50 = 15 nM T99840 C2G4DL 44446151 IC50 = 26 nM T99840 C3GDX0 44446153 IC50 = 1.6 nM T99840 C6G8RS 44446155 IC50 = 2.9 nM T99840 CO7Y2T 44446156 IC50 = 72 nM T99840 CEN64O 44446158 IC50 = 0.23 nM T99840 C0Q4XW 44446160 IC50 = 1.1 nM T99840 CMRT79 44446161 IC50 = 7.4 nM T99840 CWQ95D 44446163 IC50 = 288 nM T99840 C4S8ZQ 44446166 IC50 = 262 nM T99840 CZ3U6D 44446167 IC50 = 6.5 nM T99840 C2WQ3C 44446169 IC50 = 29 nM T99840 C71ELD 44446170 IC50 = 36 nM T99840 C6EK8F 44446171 IC50 = 50 nM T99840 C8ZK5B 44446172 IC50 = 3.1 nM T99840 C6PEY0 44446174 IC50 = 29 nM T99840 C5IW0Y 44446176 IC50 = 84 nM T99840 CMXW56 44446179 IC50 = 18 nM T99840 CNQH17 44446182 IC50 = 11 nM T99840 CK73CX 44446183 IC50 = 12 nM T99840 CPZA49 44446184 IC50 = 0.9 nM T99840 C4CZ9L 44446185 IC50 = 4.8 nM T99840 CW4Y9I 44446186 IC50 = 1.2 nM T99840 CIRM84 44446191 IC50 = 6.1 nM T99840 C5KCU2 44446192 IC50 = 61 nM T99840 CI69XS 44446193 IC50 = 0.75 nM T99840 CES2P4 44446194 IC50 = 15 nM T99840 C3MHK1 44446195 IC50 = 0.53 nM T99840 C7WKO1 44449123 IC50 = 8.7 nM T99840 CY27LD 44454961 IC50 > 10000 nM T99840 CK4BV0 44454962 IC50 = 257 nM T99840 CX5BZ2 44454988 IC50 > 10000 nM T99840 CD3QS7 44454989 IC50 = 685 nM T99840 C4BXT1 44455020 IC50 = 416 nM T99840 CT2UR5 44455050 IC50 = 212 nM T99840 CLQR53 44455051 IC50 = 105 nM T99840 CO01UH 44455052 IC50 = 81 nM T99840 CLRN39 44455054 IC50 = 62 nM T99840 CXYT35 44455355 IC50 = 23 nM T99840 CRWP10 44455388 IC50 > 10000 nM T99840 CJVC30 44455408 IC50 > 10000 nM T99840 C20GEX 44455409 IC50 > 10000 nM T99840 CO3V6X 44455431 IC50 > 10000 nM T99840 CYK50G 44455497 IC50 = 390 nM T99840 C4UK8G 44455523 IC50 = 3500 nM T99840 C8SFN2 44455525 IC50 = 2000 nM T99840 CNQ65C 44455577 IC50 = 150 nM T99840 CK75MF 44455580 IC50 = 17000 nM T99840 C8D6SZ 44455609 IC50 = 110 nM T99840 CPTW62 44455611 IC50 = 9000 nM T99840 CTW4Z5 44455643 IC50 = 150 nM T99840 C0O4PB 44455644 IC50 = 14000 nM T99840 C1C0OR 44455646 IC50 > 20000 nM T99840 CXYD92 44455729 IC50 = 30 nM T99840 C98DZW 44455731 IC50 = 8 nM T99840 CE4Q3W 44455732 IC50 = 2600 nM T99840 C2P5MJ 44455804 IC50 = 20 nM T99840 CQS0H9 44455828 IC50 > 20000 nM T99840 C85CZH 44571533 IC50 = 0.7 nM T99840 C24IJZ 44571534 IC50 = 0.6 nM T99840 CT0Z2K 44626366 IC50 > 50000 nM T99840 CI1G4L 44814464 IC50 = 13000 nM T99840 CJG7H3 44815008 IC50 = 22000 nM T99840 CGEF05 45101437 IC50 = 0.67 nM T99840 CW5DH0 45263545 IC50 = 3 nM T99840 CZP0C2 45263546 IC50 = 83 nM T99840 CFA23Y 45263651 IC50 = 0.8 nM T99840 C79OBA 45263654 IC50 = 7.9 nM T99840 C19VMP 45279238 IC50 = 0.75 nM T99840 CAI2S3 45279243 IC50 = 4 nM T99840 CVE8H0 45279329 IC50 = 32 nM T99840 CMU1Y2 45279330 IC50 = 20 nM T99840 C98ZUP 45279331 IC50 = 175 nM T99840 CNL75F 45279417 IC50 = 94 nM T99840 CO4ZS2 45279505 IC50 = 26 nM T99840 CY3H1B 45279506 IC50 = 1 nM T99840 CVE91H 45279510 IC50 = 10 nM T99840 C1IT0C 45279600 IC50 = 2229 nM T99840 CXU8W7 45485422 IC50 = 2.9 nM T99840 C64YKE 45485436 IC50 = 4.2 nM T99840 C8Q0FP 45485446 IC50 = 3.2 nM T99840 CG2JD6 45485450 IC50 = 0.31 nM T99840 CM3DO4 45485456 IC50 = 0.37 nM T99840 CAO31T 45485464 IC50 = 0.41 nM T99840 C8JES7 45485471 IC50 = 0.58 nM T99840 C5UBN2 45485490 IC50 = 1.5 nM T99840 CZU9L2 45485491 IC50 = 0.2 nM T99840 CK6ZT7 45485492 IC50 = 0.62 nM T99840 CJ6TP3 45485495 IC50 = 0.26 nM T99840 CR2FZ0 45485496 IC50 = 0.44 nM T99840 CEWX31 45485523 IC50 = 0.17 nM T99840 COU45W 45485527 IC50 = 0.26 nM T99840 CV9W4F 45485533 IC50 = 0.26 nM T99840 CIWV94 45485553 IC50 = 0.24 nM T99840 CDZ84U 45487083 IC50 = 2510 nM T99840 CP7O3K 45487084 IC50 = 4889 nM T99840 CMH59T 45487090 IC50 = 5722 nM T99840 CN86WT 45487093 IC50 = 0.52 nM T99840 CK8J0C 45487094 IC50 = 66 nM T99840 C9WD4X 45487096 IC50 = 202 nM T99840 C6Q5MP 45487102 IC50 = 678 nM T99840 CS20OB 45487103 IC50 = 1109 nM T99840 C29SDN 45487104 IC50 = 70 nM T99840 C5EO7Y 45487109 IC50 = 989 nM T99840 CA8BF4 45487115 IC50 = 8813 nM T99840 CU90YF 45487122 IC50 = 9 nM T99840 CH0N3P 45487123 IC50 = 194 nM T99840 C4EU3H 45487124 IC50 = 2 nM T99840 CAP86G 45487130 IC50 = 1066 nM T99840 C5RJ4D 45487131 IC50 = 826 nM T99840 CGVJ06 45487146 IC50 = 1 nM T99840 CGUL09 45487151 IC50 = 5654 nM T99840 CUC2W8 46186977 EC50 = 47600 nM T99840 CE9U3O 46189877 IC50 = 13300 nM T99840 CN8C1E 46200343 IC50 = 191 nM T99840 C92RAS 46200344 IC50 = 72 nM T99840 CDK02H 46201982 IC50 = 230 nM T99840 CRLM46 46201983 IC50 = 33 nM T99840 CXAK48 46203600 IC50 = 300 nM T99840 C40JBU 46203602 IC50 = 76 nM T99840 CMG2U0 46204901 IC50 = 87 nM T99840 CTXE90 46205227 IC50 = 37 nM T99840 C6UNV9 46205555 IC50 = 56 nM T99840 CLG92T 46205556 IC50 = 5400 nM T99840 CK1ZG6 46205872 IC50 = 44 nM T99840 C8ONI5 46205873 IC50 = 1900 nM T99840 CFO2S8 46205876 IC50 = 19000 nM T99840 CS7A1F 46206542 IC50 = 530 nM T99840 C64UTP 46206544 IC50 = 3100 nM T99840 CVW24X 46206545 IC50 = 80 nM T99840 CN7QE6 46206546 IC50 = 100 nM T99840 C4K3DZ 46206874 IC50 = 3300 nM T99840 CJ79UT 46206875 IC50 = 120 nM T99840 CYP2H6 46206879 IC50 = 820 nM T99840 CK4TI1 46214177 IC50 = 130 nM T99840 CE02DJ 46214505 IC50 = 1260 nM T99840 CQ5G0O 46214506 IC50 = 37 nM T99840 CQ1Z0D 46214507 IC50 = 140 nM T99840 CPF0J9 46214673 IC50 = 39 nM T99840 CV2Q4F 46214674 IC50 = 49 nM T99840 CEB7L5 46214832 IC50 = 35 nM T99840 C8KE9V 46214983 IC50 = 2500 nM T99840 C5TEA2 46214986 IC50 = 1100 nM T99840 CME1P7 46215156 IC50 = 24 nM T99840 CX5BE1 46215326 IC50 = 16 nM T99840 CL58QM 46215511 IC50 = 40 nM T99840 C0QS3H 46215512 IC50 = 95 nM T99840 C35ZCM 46215514 IC50 = 240 nM T99840 C5DV7T 46216355 IC50 = 41 nM T99840 CT6J2S 46216529 IC50 = 41 nM T99840 CL86HB 46216678 EC50 = 501.19 nM T99840 CX7K3M 46216736 IC50 = 6140 nM T99840 C83ZQU 46225338 IC50 > 10000 nM T99840 CN74XF 46225339 IC50 = 390 nM T99840 C43PME 46225360 IC50 = 600 nM T99840 C12LPT 46225361 IC50 = 640 nM T99840 C8A3DL 46228934 IC50 > 30000 nM T99840 CR4KT7 46229901 IC50 > 50000 nM T99840 CW4P2I 46229902 IC50 > 50000 nM T99840 C5FB9H 46229972 IC50 > 50000 nM T99840 C9L8MQ 46229973 IC50 > 50000 nM T99840 CJAH09 46229974 IC50 = 34430 nM T99840 COFP27 46231466 IC50 = 1995.26 nM T99840 CD7CJ3 46231467 IC50 = 10000 nM T99840 C86UDB 46231469 EC50 = 10000 nM T99840 CPJ4R8 46231471 IC50 = 1000 nM T99840 C19JAS 46231522 IC50 = 630.96 nM T99840 CMF8X1 46231524 IC50 = 630.96 nM T99840 CFAK81 46231526 IC50 = 251.19 nM T99840 C1G9YE 46231528 IC50 = 1258.93 nM T99840 CP9Y1S 46231577 EC50 = 501.19 nM T99840 CS2EI9 46231579 IC50 = 10000 nM T99840 C4U6HW 46231628 IC50 = 25118.86 nM T99840 CNH5D1 46231630 IC50 = 1258.93 nM T99840 CC03FA 46231632 IC50 = 1584.89 nM T99840 C7XNM1 46231634 IC50 = 1995.26 nM T99840 CUPG59 46231688 IC50 = 316.23 nM T99840 C2GIB6 46231690 IC50 = 1258.93 nM T99840 COA9P3 46231692 IC50 = 398.11 nM T99840 C5H0AL 46231694 IC50 = 794.33 nM T99840 CZ36XF 46231747 IC50 = 398.11 nM T99840 CSA40G 46231749 IC50 = 794.33 nM T99840 CH0CA1 46231751 IC50 = 1258.93 nM T99840 C0XBY7 46231753 IC50 = 630.96 nM T99840 CDA42Z 46231821 IC50 = 12589.25 nM T99840 CKT0W9 46236732 IC50 = 0.35 nM T99840 CP4L1C 46236733 IC50 = 250 nM T99840 CO0QT7 46841575 IC50 = 26 nM T99840 CO31WX 46861576 IC50 = 16 nM T99840 C8EX6T 46864718 EC50 = 6 nM T99840 CT5A7F 46871758 IC50 = 54 nM T99840 CIS65O 46871825 IC50 = 1.9 nM T99840 C5Y2ZB 46878651 EC50 = 1400 nM T99840 C3UO4V 46878691 EC50 = 9300 nM T99840 CBEO79 46878692 EC50 = 12600 nM T99840 C3JCD4 46878693 EC50 = 9200 nM T99840 CH3Y9O 46878694 EC50 > 40000 nM T99840 CUK40A 46878737 EC50 = 7600 nM T99840 C2Z9UW 46878738 EC50 > 80000 nM T99840 CWA51E 46878739 EC50 > 80000 nM T99840 C41OTL 46878740 EC50 = 16100 nM T99840 CT1N2L 46878785 EC50 > 40000 nM T99840 CI23FY 46878786 IC50 = 36100 nM T99840 CS6N2R 46878787 EC50 > 40000 nM T99840 CEN9Y3 46878788 EC50 > 40000 nM T99840 CR1ZX3 46878848 EC50 > 80000 nM T99840 CFRJ50 46878849 EC50 > 80000 nM T99840 C5WXJ0 46878850 EC50 > 40000 nM T99840 CC29YQ 46878851 EC50 > 40000 nM T99840 C9GAN2 46878852 EC50 = 47600 nM T99840 C7VA3G 46883541 IC50 = 2.1 nM T99840 CRAO48 46883741 IC50 = 5000 nM T99840 CFI6X4 46883745 IC50 = 20 nM T99840 C3DSI2 46883776 IC50 = 651 nM T99840 CP8Q6Y 46883777 IC50 = 467 nM T99840 CCPX03 46883778 IC50 = 6 nM T99840 COZ41D 46883779 IC50 = 1 nM T99840 C8S7FD 46883804 IC50 = 0.77 nM T99840 CF82LP 46884323 IC50 = 1698 nM T99840 CD50RE 46884324 IC50 = 760 nM T99840 CEW94S 46884370 IC50 = 662 nM T99840 C2YZ8W 46884456 IC50 = 557 nM T99840 CNH6Y3 46884457 IC50 = 1.01 nM T99840 CA67FX 46884483 IC50 = 3.7 nM T99840 CY0G3Q 46884484 IC50 = 22.4 nM T99840 CB7MI5 46884678 IC50 = 9200 nM T99840 COW3L9 46884679 IC50 > 50000 nM T99840 CM78KJ 46884705 IC50 > 50000 nM T99840 CJG0C1 46884792 IC50 = 9100 nM T99840 C1MP7S 46890758 IC50 = 25072 nM T99840 CEW8I9 46890759 IC50 = 187 nM T99840 CT5KD7 46890760 IC50 = 71 nM T99840 C6UBC0 46890761 IC50 = 574 nM T99840 CU20TA 46890816 IC50 = 418 nM T99840 C40CHX 46890817 IC50 = 358 nM T99840 CX9KP3 46890818 IC50 = 771 nM T99840 C9HBP7 46890819 IC50 = 304 nM T99840 CI6SX2 46890820 IC50 = 403 nM T99840 C8YU2V 46890880 IC50 = 304 nM T99840 CY6BV2 46890881 IC50 = 138 nM T99840 C5J8IW 46890882 IC50 = 34 nM T99840 C6CXV3 46890883 IC50 = 13 nM T99840 CKW2T8 46890943 IC50 = 2656 nM T99840 CCH1L9 46890944 IC50 = 995 nM T99840 CXO39V 46890945 IC50 = 235 nM T99840 C9LPA4 46891002 IC50 = 6209 nM T99840 CL47FR 46891003 IC50 = 576 nM T99840 C4VWG2 46891052 IC50 = 25 nM T99840 CMGW50 46891411 IC50 = 546 nM T99840 C6EA2X 46891412 IC50 = 288 nM T99840 CRBX43 46891413 IC50 > 40000 nM T99840 C24XZM 46891455 IC50 > 40000 nM T99840 CRAM45 46891456 IC50 > 40000 nM T99840 CNAX47 46891457 IC50 > 40000 nM T99840 CBL1E2 46891458 IC50 > 40000 nM T99840 CN4RS8 46891517 IC50 = 2302 nM T99840 C2C3LG 46891518 IC50 = 2792 nM T99840 C9R5UL 46891519 IC50 > 40000 nM T99840 CF12WN 46891520 IC50 > 40000 nM T99840 C1B8DK 46891521 IC50 = 18334 nM T99840 C15OSQ 46891575 IC50 > 40000 nM T99840 CLO7S1 46891576 IC50 > 40000 nM T99840 C61NMK 46891577 IC50 = 4000 nM T99840 CZ8V9I 46891578 IC50 = 2361 nM T99840 C4KNU1 46891579 IC50 = 6704 nM T99840 CZ7C1J 46893145 IC50 = 130 nM T99840 CP2FI0 46912223 IC50 = 1.7 nM T99840 CF35QN 49865652 IC50 = 3502 nM T99840 CYNH04 49865736 IC50 = 229 nM T99840 CW2M9C 49865787 IC50 = 7100 nM T99840 CD49WA 49865788 IC50 = 106 nM T99840 C79LFV 49865865 IC50 = 85 nM T99840 C3J7YR 49865866 IC50 = 503 nM T99840 CWX5Y7 49865867 IC50 = 73 nM T99840 CED86P 49865925 IC50 > 20000 nM T99840 CL3K5Q 49865926 IC50 > 20 nM T99840 C4Z0BG 49866251 IC50 = 163 nM T99840 C7GR0H 49872381 IC50 = 40 nM T99840 CD1X3U 49872384 IC50 = 28 nM T99840 C6B0NT 49872385 IC50 = 60 nM T99840 CZML42 49872482 IC50 = 68 nM T99840 C60RMP 49872483 IC50 = 19 nM T99840 CA3QJ9 50898349 IC50 = 122 nM T99840 CZIS04 50899302 IC50 = 900 nM T99840 C4BD6H 52935148 IC50 = 158 nM T99840 C3Q6TV 52939724 IC50 = 200 nM T99840 CF86AB 52946557 IC50 = 800 nM T99840 CBS28G 52947827 IC50 = 1400 nM T99840 CTV15R 52949026 IC50 = 1500 nM T99840 CWQ8Y2 53307787 IC50 = 300 nM T99840 CR7TD8 53307788 IC50 = 200 nM T99840 C8XR3L 53316726 IC50 = 342 nM T99840 CVY45A 53316727 IC50 = 19316 nM T99840 C1SBC9 53316728 IC50 = 1919 nM T99840 CR3E5C 53316729 IC50 = 448 nM T99840 CU72TL 53316730 IC50 = 164 nM T99840 C9RK8W 53317504 IC50 = 1860 nM T99840 CXT58Z 53318019 IC50 = 20000 nM T99840 C37ZAQ 53318697 IC50 = 370 nM T99840 CBLD50 53318698 IC50 = 200 nM T99840 CIN82X 53319361 IC50 = 537 nM T99840 C68CRW 53319362 IC50 = 356 nM T99840 C5YZC0 53319363 IC50 = 440 nM T99840 C8U2PO 53319364 IC50 = 875 nM T99840 CC37JA 53319365 IC50 = 935 nM T99840 CM4H0Y 53319366 IC50 = 209 nM T99840 CUG7V3 53320013 IC50 = 2080 nM T99840 CS04NZ 53320014 IC50 = 1070 nM T99840 CKJQ81 53320673 IC50 = 156 nM T99840 C0SU6P 53320674 IC50 = 2531 nM T99840 CMG8J3 53320675 IC50 = 1409 nM T99840 CQD62W 53321323 IC50 = 540 nM T99840 COT69M 53321324 IC50 = 320 nM T99840 CJO8K6 53321365 IC50 = 1406 nM T99840 C92ZPY 53321966 IC50 = 126 nM T99840 CUP16W 53321967 IC50 = 1392 nM T99840 C4O6RY 53323317 IC50 = 145 nM T99840 CJT3O4 53323318 IC50 = 16374 nM T99840 CT0IN8 53323319 IC50 = 485 nM T99840 CMG85A 53323320 IC50 = 465 nM T99840 C5RDB1 53323321 IC50 = 540 nM T99840 C8ZHY7 53323979 IC50 > 10000 nM T99840 C9Q1ND 53324647 IC50 = 20000 nM T99840 CV9XG0 53324648 IC50 = 2069 nM T99840 CB35NA 53324649 IC50 = 2215 nM T99840 C2FV4W 53324650 IC50 = 201 nM T99840 CUO1R8 53325274 IC50 = 1290 nM T99840 CZB7M2 53325275 IC50 = 1690 nM T99840 CLV49B 53325838 IC50 = 649 nM T99840 C7GQK5 53325949 IC50 = 552 nM T99840 C3KWC5 53326627 IC50 = 1650 nM T99840 CZ8DU9 53326926 IC50 = 619 nM T99840 CF67UL 53327840 IC50 = 0.4 nM T99840 C6ACY1 53466872 IC50 > 4000 nM T99840 C4U5IX 53493001 EC50 = 70 nM T99840 CMNA20 54580854 IC50 = 2.7 nM T99840 C46ZWI 54580879 IC50 = 1.7 nM T99840 CD45JK 54581914 IC50 = 263 nM T99840 C6EPJ0 54581915 IC50 = 82.8 nM T99840 CTCM02 54581934 IC50 = 226 nM T99840 C50EXN 54581935 IC50 = 0.8 nM T99840 C5RDG6 54581936 IC50 > 10000 nM T99840 CJ1WZ3 54582829 IC50 = 52.7 nM T99840 C94LQC 54582858 IC50 = 7.8 nM T99840 C3QVP4 54582859 IC50 = 9.4 nM T99840 CRAW75 54582860 IC50 = 3100 nM T99840 CHX16Y 54582861 IC50 = 250 nM T99840 CIKC16 54582862 IC50 = 480 nM T99840 CZ4DV0 54582863 IC50 = 8.9 nM T99840 CY81FK 54582864 IC50 = 5.4 nM T99840 CUL04M 54583866 IC50 = 21.6 nM T99840 CA3UH9 54583867 IC50 = 31 nM T99840 C0O8UB 54583868 IC50 = 2.9 nM T99840 CIT94F 54583869 IC50 = 3.3 nM T99840 CFO6L2 54583870 IC50 = 4.6 nM T99840 CFL7C6 54584820 IC50 = 2.5 nM T99840 CTO6N3 54584821 IC50 = 148 nM T99840 CZ5IA1 54585612 IC50 = 3.8 nM T99840 CZR3A2 54585748 IC50 = 0.39 nM T99840 CQH3O5 54585770 IC50 = 64.6 nM T99840 C0W3NV 54585771 IC50 = 310 nM T99840 CM45DH 54585772 IC50 = 19.5 nM T99840 CJM86T 54585773 IC50 = 19.3 nM T99840 CM6KH7 54585774 IC50 = 6.9 nM T99840 CCK9Z3 54586727 IC50 = 14.6 nM T99840 C8TMD3 54586758 IC50 = 3.6 nM T99840 C2G0RU 54586759 IC50 = 4.3 nM T99840 CV1L4K 54586760 IC50 = 8.2 nM T99840 C6L0WH 54586761 IC50 = 4.9 nM T99840 CYT89D 54587765 IC50 = 1.2 nM T99840 CE19HM 54587781 IC50 = 0.4 nM T99840 C5GC3J 54587782 IC50 = 45.7 nM T99840 C8NYA1 54587783 IC50 = 7.9 nM T99840 C0AIO8 54587784 IC50 = 53.9 nM T99840 CNA7I0 54587785 IC50 = 93.3 nM T99840 C0VYX8 54669875 IC50 = 7.99 nM T99840 C24UKQ 54764004 IC50 = 125.89 nM T99840 C9LF2N 56592447 EC50 = 30 nM T99840 CQ1GO6 56658871 IC50 = 10457 nM T99840 CE05WK 56658872 IC50 = 8 nM T99840 CTKA80 56659252 EC50 = 21000 nM T99840 CI48MU 56659253 EC50 = 19000 nM T99840 C3TAV6 56659254 EC50 = 49000 nM T99840 C4KGE6 56659627 IC50 = 794.33 nM T99840 CXZW56 56659628 IC50 > 100000 nM T99840 CS4N2M 56659870 IC50 = 1640 nM T99840 CI1Z4B 56659871 IC50 = 1000 nM T99840 C0PSG1 56659872 IC50 = 270 nM T99840 C2RX1T 56662356 IC50 = 187 nM T99840 CWS15Q 56662733 IC50 = 12900 nM T99840 CU25CK 56662734 IC50 = 89000 nM T99840 CXSD38 56663088 IC50 = 316.23 nM T99840 CB9ZN5 56663089 IC50 = 50118.72 nM T99840 C1IPX6 56663090 IC50 = 1995.26 nM T99840 CN70JC 56663117 IC50 = 316.23 nM T99840 CK5FY6 56663118 IC50 = 100 nM T99840 CXE41B 56663331 IC50 = 7060 nM T99840 C0PTB8 56663332 IC50 = 7010 nM T99840 CU6NX4 56665650 IC50 = 29 nM T99840 CV04XS 56666134 IC50 > 500 nM T99840 CJ8AQ3 56666135 IC50 > 80000 nM T99840 CZE94O 56666199 IC50 = 32000 nM T99840 C01YFA 56666200 IC50 > 80000 nM T99840 C9SC6L 56666757 IC50 = 5710 nM T99840 C4MFS5 56666758 IC50 = 450 nM T99840 CF0KZ2 56666759 IC50 = 820 nM T99840 C62JDU 56666760 IC50 = 410 nM T99840 C1GH7Y 56669242 IC50 = 18719 nM T99840 C1P6WA 56669243 IC50 = 29 nM T99840 CK71EP 56669244 IC50 = 888 nM T99840 C5D7ZT 56669536 EC50 = 12000 nM T99840 C2F4UM 56669537 EC50 = 8000 nM T99840 CA1ME9 56669597 IC50 = 80000 nM T99840 CP8M7G 56669598 IC50 = 27000 nM T99840 C25AQX 56669599 IC50 > 80000 nM T99840 C3L4ZK 56669956 IC50 = 10000 nM T99840 C06PUJ 56669957 IC50 = 501.19 nM T99840 C3U4AP 56669979 IC50 = 79.43 nM T99840 C78SDI 56669980 IC50 = 158.49 nM T99840 CZO49F 56670192 IC50 = 2640 nM T99840 CJ8P3S 56672571 IC50 = 21 nM T99840 C3GV1C 56672708 IC50 = 4 nM T99840 CTD9Z3 56672709 IC50 = 4 nM T99840 C8WG2N 56672710 IC50 = 767 nM T99840 CNR2P1 56673049 EC50 = 21000 nM T99840 C7C4VZ 56673050 EC50 = 32000 nM T99840 CPUK68 56673051 EC50 > 80000 nM T99840 CS7KW0 56673052 IC50 > 80000 nM T99840 CCQK10 56673053 IC50 = 102000 nM T99840 CZPU76 56673054 EC50 > 40000 nM T99840 CE78CJ 56673118 IC50 = 104000 nM T99840 CI8P9J 56673119 EC50 = 15000 nM T99840 CXM90K 56673464 IC50 = 6309.57 nM T99840 C2GN9F 56673465 IC50 = 3162.28 nM T99840 CL0Q3N 56673466 IC50 = 398.11 nM T99840 C7E3IP 56673494 IC50 = 100 nM T99840 CL4P9H 56673495 IC50 = 50.12 nM T99840 C4G0YE 56673715 IC50 = 1220 nM T99840 CWZV47 56673716 IC50 = 220 nM T99840 C1KW9Z 56673717 IC50 = 4040 nM T99840 CJUC47 56676069 IC50 = 7 nM T99840 CQV4B5 56676365 IC50 = 105000 nM T99840 CN81GL 56676366 EC50 = 21000 nM T99840 C9YV7U 56676367 EC50 > 10000 nM T99840 C6DAW2 56676435 IC50 = 31000 nM T99840 C6KCR5 56676736 IC50 = 79.43 nM T99840 C70DIW 56676779 IC50 = 199.53 nM T99840 C4KL0A 56676780 IC50 = 5011.87 nM T99840 C79ILY 56677020 IC50 = 1940 nM T99840 CL7AW3 56677021 IC50 = 780 nM T99840 CVXN71 56679251 IC50 = 14 nM T99840 CUHO31 56679252 IC50 = 16 nM T99840 C82YOE 56679400 IC50 = 28 nM T99840 C0C3TN 56679401 IC50 = 437 nM T99840 C7YM2G 56679402 IC50 = 149 nM T99840 C7QRM2 56679701 EC50 = 50000 nM T99840 CZO95E 56679702 IC50 = 24000 nM T99840 C4VU6Z 56679703 IC50 > 40000 nM T99840 C4LO5Q 56679704 IC50 > 80000 nM T99840 CQ8K7M 56680096 IC50 = 398.11 nM T99840 C6EO3N 56680128 IC50 = 39.81 nM T99840 C2KEV0 56680350 IC50 > 10000 nM T99840 C9DTH0 56680351 IC50 = 490 nM T99840 CMR0J9 56680352 IC50 = 1410 nM T99840 CDXT81 56681654 IC50 = 270 nM T99840 CYZ34G 56682694 IC50 = 22 nM T99840 C13LZJ 56683026 EC50 = 23000 nM T99840 CTC48A 56683027 EC50 > 80000 nM T99840 CVR0H1 56683437 IC50 = 251.19 nM T99840 CR8N0J 56683438 IC50 = 10000 nM T99840 C24XYT 56683439 IC50 = 251.19 nM T99840 C2MJ4D 56683476 IC50 = 2511.89 nM T99840 CKF29M 56683680 IC50 > 10000 nM T99840 C4X7IP 56683681 IC50 = 1440 nM T99840 C18ADK 56833940 IC50 = 16.9 nM T99840 C1MFZ4 56833941 IC50 = 16.5 nM T99840 C3I9PO 56833942 IC50 = 72.4 nM T99840 CHC9A6 56833943 IC50 = 49 nM T99840 CD30YZ 56833944 IC50 = 49.5 nM T99840 CO3EV9 56833945 IC50 = 12.3 nM T99840 CT16AO 56834043 IC50 = 16.6 nM T99840 CMI5T6 56834044 IC50 = 11.7 nM T99840 CCNF23 56834045 IC50 = 7.97 nM T99840 CMOU39 56834046 IC50 = 27.9 nM T99840 C4LQM9 56834047 IC50 = 33.8 nM T99840 CCP0K8 56834048 IC50 = 45.2 nM T99840 CP0VQ2 56834146 IC50 = 8.58 nM T99840 CMPT46 56834147 IC50 = 5.25 nM T99840 CD0K6U 56834148 IC50 = 7.53 nM T99840 CTDB01 56834149 IC50 = 13.4 nM T99840 CK4RN1 56834150 IC50 = 11.2 nM T99840 CP82BX 56834151 IC50 = 5.51 nM T99840 C6I8SK 56834259 IC50 = 44.5 nM T99840 CSCR53 56834260 IC50 = 16.4 nM T99840 CO6L5V 56834261 IC50 = 10.8 nM T99840 CJY10S 56834262 IC50 = 6.46 nM T99840 CQ84ZA 56945122 EC50 = 29 nM T99840 C0WBY6 56945991 IC50 = 187 nM T99840 C87GZI 56946207 IC50 = 122 nM T99840 C6A2FU 56946208 IC50 = 18833 nM T99840 CMAU62 56946312 IC50 = 80 nM T99840 C2E5TO 56946313 IC50 = 199 nM T99840 CHRU78 56946423 IC50 = 29 nM T99840 CQB9G8 56946424 IC50 = 7643 nM T99840 CI28DU 56946526 IC50 = 16237 nM T99840 C4MDZ6 56946527 IC50 = 89 nM T99840 C1KI4X 56946528 IC50 = 3210 nM T99840 C52OXA 56946529 IC50 = 26 nM T99840 CKM18B 56946627 IC50 = 53 nM T99840 CQ2MT0 56946628 IC50 = 117 nM T99840 CDQN37 56946629 IC50 = 21 nM T99840 C5VIB3 56946630 IC50 = 103 nM T99840 CSE28N 56946631 IC50 = 106 nM T99840 CE68HR 56953105 IC50 = 1.77 nM T99840 CJ3O9S 57327010 IC50 = 0.27 nM T99840 CYCP25 57327180 IC50 = 0.178 nM T99840 C30IZU 57384527 IC50 = 0.99 nM T99840 CQA35K 57384528 IC50 = 22.5 nM T99840 CJ3C9M 57384790 IC50 = 87.1 nM T99840 CGL94D 57384791 IC50 = 11.1 nM T99840 CMJ10O 57384792 IC50 = 6.92 nM T99840 C3MP2C 57384793 IC50 = 14.7 nM T99840 C0X1DZ 57384794 IC50 = 4.77 nM T99840 CN0YS7 57385030 IC50 = 7.47 nM T99840 CF5D1K 57385031 IC50 = 9.6 nM T99840 CEH5V4 57385032 IC50 = 4.11 nM T99840 C9LM2N 57385033 IC50 = 24.4 nM T99840 CSA8N6 57385034 IC50 = 12.1 nM T99840 CWZY54 57385280 IC50 = 45.5 nM T99840 CRO35Q 57385281 IC50 = 12.3 nM T99840 CMDX46 57390296 IC50 > 1250 nM T99840 C97PNB 57390896 IC50 = 56 nM T99840 CL2C3I 57392070 IC50 = 52 nM T99840 CX7L1C 57392134 IC50 = 2868 nM T99840 CRXD10 57392696 IC50 = 60 nM T99840 C5IM8F 57393826 IC50 = 3431 nM T99840 CHET54 57393827 IC50 = 3358 nM T99840 CJIZ48 57397373 IC50 = 999 nM T99840 CH32BO 57397434 IC50 > 5000 nM T99840 CO14BW 57397444 IC50 = 376 nM T99840 CVRD17 57399109 IC50 > 40000 nM T99840 CZLD01 57399119 IC50 = 5548 nM T99840 CW2DO9 57399120 IC50 = 483 nM T99840 CG7NW9 57400793 IC50 = 675 nM T99840 CR6AE3 57400851 EC50 = 1500 nM T99840 CYVN84 57402550 IC50 = 733 nM T99840 C5XF1Z 57402551 IC50 = 86 nM T99840 CSCH73 57404337 IC50 > 50000 nM T99840 C4QT2R 57404351 IC50 = 1000 nM T99840 CS1V8U 57404352 IC50 = 4 nM T99840 CKU6E8 57404500 IC50 > 50000 nM T99840 CXHN06 57987388 IC50 = 120 nM T99840 CXW7P5 58063504 IC50 = 18 nM T99840 C1XI2O 58063517 IC50 = 145 nM T99840 CEWR70 58065681 IC50 = 183 nM T99840 C15MAW 58065745 IC50 = 17 nM T99840 CRZH72 58173522 IC50 = 120 nM T99840 CGTB71 58445369 IC50 = 250 nM T99840 C0IZ4O 58469132 IC50 > 20000 nM T99840 CE94VP 58528692 IC50 = 210 nM T99840 CR4GK2 58528697 IC50 = 83 nM T99840 C1JO3I 58528715 IC50 = 9000 nM T99840 CH83XK 58528726 IC50 = 250 nM T99840 C5R7ZG 58528729 IC50 = 130 nM T99840 CS8WO1 58528732 IC50 = 39 nM T99840 CX3SQ7 58528738 IC50 = 88 nM T99840 CZEK86 58528741 IC50 = 140 nM T99840 C0VL2K 58528743 IC50 = 1500 nM T99840 CU2G9R 58528758 IC50 = 73 nM T99840 CY9SH8 58528759 IC50 = 400 nM T99840 C54KGY 58528775 IC50 = 580 nM T99840 C70BOM 58528779 IC50 = 3700 nM T99840 CLE51O 58528784 IC50 = 6700 nM T99840 C6P8SD 58548876 IC50 = 52 nM T99840 C0N5GT 58850279 IC50 = 4 nM T99840 C83YXM 58910631 IC50 = 130 nM T99840 CP91WC 58910757 EC50 = 1500 nM T99840 CG3Y5M 58950709 IC50 = 6.8 nM T99840 CVBT13 59201219 IC50 = 45 nM T99840 C1E3XT 59472470 IC50 = 42 nM T99840 C92NPY 59472493 IC50 = 1250 nM T99840 CL4F1U 59472507 IC50 = 8710 nM T99840 CG1ZH6 59472511 IC50 = 3980 nM T99840 CHU2S4 59472516 IC50 = 200 nM T99840 CW4I0H 59472517 IC50 = 40 nM T99840 C4RZ7E 59472522 IC50 = 390 nM T99840 CKS31U 59472524 IC50 = 180 nM T99840 C35EKB 59472530 IC50 = 10 nM T99840 CLB40A 59472544 IC50 = 78 nM T99840 CL9Y0P 59472546 IC50 = 680 nM T99840 CXH19J 59472574 IC50 = 30 nM T99840 C51KUS 59472588 IC50 = 70 nM T99840 CPH07V 59472599 IC50 = 78 nM T99840 CS87XI 59472603 IC50 = 150 nM T99840 CI8H4T 59472630 IC50 = 1630 nM T99840 CXO21N 59472637 IC50 = 3860 nM T99840 CH0S6A 59472641 IC50 = 430 nM T99840 C0LBN5 59472644 IC50 = 4850 nM T99840 C4SR9V 59472646 IC50 = 1270 nM T99840 C6D7LS 59472679 IC50 = 160 nM T99840 C8UMR6 59472684 IC50 = 40 nM T99840 C1ME7D 59472698 IC50 = 2010 nM T99840 CYO06N 59472699 IC50 = 370 nM T99840 C6XDH2 59472707 IC50 = 90 nM T99840 CF72WU 59472713 IC50 = 440 nM T99840 C9L0GJ 59472717 IC50 = 4420 nM T99840 CGD8W0 59472725 IC50 = 38 nM T99840 C2T4EU 59472735 IC50 = 380 nM T99840 CJR3K7 59472756 IC50 = 180 nM T99840 C1RUN6 59472765 IC50 = 70 nM T99840 CZ52KP 59472771 IC50 = 940 nM T99840 CB3X0F 59472773 IC50 = 1080 nM T99840 C6YZR8 59472775 IC50 = 480 nM T99840 CDOV85 59472789 IC50 = 1110 nM T99840 CWD0K3 59472815 IC50 = 270 nM T99840 C05YQD 59472822 IC50 = 28 nM T99840 C15JGP 59472849 IC50 = 1190 nM T99840 CM0G7S 59472858 IC50 = 940 nM T99840 CEP94I 59472861 IC50 = 80 nM T99840 CLH47W 59472872 IC50 = 150 nM T99840 CKGD30 59570713 IC50 > 100000 nM T99840 C18TXZ 60150510 IC50 = 10 nM T99840 C30UIB 60150707 IC50 = 9 nM T99840 C3V4UC 66549618 IC50 > 5000 nM T99840 CM4QT6 66551384 IC50 = 18 nM T99840 CO27HW 66551578 IC50 = 17 nM T99840 CZX69Y 66551579 IC50 = 25 nM T99840 CY7XR2 66551580 IC50 = 59 nM T99840 CPGZ81 66551772 IC50 = 30 nM T99840 CSP8G3 66678794 IC50 = 145 nM T99840 C9VW4M 66679082 IC50 = 25 nM T99840 CF6X2S 66679323 IC50 = 43 nM T99840 CK1J6R 66679335 IC50 = 69 nM T99840 C96BLD 66679340 IC50 = 5289 nM T99840 C79GQM 66679372 IC50 = 107 nM T99840 C8LMK0 66679376 IC50 = 2113 nM T99840 CZKV14 66679405 IC50 = 17 nM T99840 CYEL45 66679447 IC50 = 82 nM T99840 C1CUA9 66679503 IC50 = 696 nM T99840 CJ0KL5 66679507 IC50 = 73 nM T99840 C9RS5B 66679618 IC50 = 94 nM T99840 CXN25J 66679626 IC50 = 203 nM T99840 CG5W9J 66679630 IC50 = 1660 nM T99840 C39KZH 66679674 IC50 = 592 nM T99840 CUC7E1 66679703 IC50 = 60 nM T99840 C9VK6Q 66679957 IC50 = 603 nM T99840 C5LTS2 66790999 IC50 = 420 nM T99840 C4DRN2 66791090 IC50 = 660 nM T99840 C0BM4Q 66855521 IC50 = 93 nM T99840 C41HEV 66855843 IC50 = 25 nM T99840 C95TOQ 66855889 IC50 = 447 nM T99840 CGLH60 66856047 IC50 = 270 nM T99840 C74OTM 66856571 IC50 = 5750 nM T99840 C4FE1H 66856796 IC50 = 220 nM T99840 C9LR2W 66856924 IC50 = 6920 nM T99840 C28GNT 66857307 IC50 = 190 nM T99840 CO1IU0 66857459 IC50 = 6170 nM T99840 CE3GP6 66857489 IC50 = 620 nM T99840 CRA3U4 66857678 IC50 = 650 nM T99840 CH79EA 66857904 IC50 = 120 nM T99840 CYPW36 66978859 IC50 = 130 nM T99840 CV4RP5 67281831 IC50 = 69 nM T99840 CXD91K 67282190 IC50 = 363 nM T99840 C7NYX0 67282874 IC50 = 131 nM T99840 C4RH1Q 67282977 IC50 = 133 nM T99840 CMJE32 67282979 IC50 = 18 nM T99840 CK58YL 67283019 IC50 = 2252 nM T99840 C1VB4O 67307922 IC50 > 10000 nM T99840 C48TLF 67308147 IC50 = 930 nM T99840 C52TWL 67308180 IC50 = 70 nM T99840 C5UA6K 67308257 IC50 = 140 nM T99840 CJI01M 67308518 IC50 = 180 nM T99840 C36HRD 67308603 IC50 = 31 nM T99840 CFWV49 67309019 IC50 = 220 nM T99840 C3PV1C 67309038 IC50 = 70 nM T99840 CXEF86 67309051 IC50 = 490 nM T99840 C3UAX0 67309119 IC50 = 1050 nM T99840 C2QA5E 67309143 IC50 = 540 nM T99840 C3RMS8 67309187 IC50 = 120 nM T99840 C8Z3ES 67309205 IC50 = 160 nM T99840 CC4I2B 67309244 IC50 = 170 nM T99840 CU8VA0 67309278 IC50 = 6000 nM T99840 C2NIO8 67309280 IC50 = 660 nM T99840 C7D6AF 67309490 IC50 = 4800 nM T99840 CASD21 67413813 IC50 = 138 nM T99840 CLV4R7 67414480 IC50 = 1216 nM T99840 CP9FJ2 67414954 IC50 = 194 nM T99840 C3G1ZI 67415170 IC50 = 182 nM T99840 CL8FT1 67415210 IC50 = 813 nM T99840 C9K6IY 67415502 IC50 = 339 nM T99840 C4GSO6 67415529 IC50 = 26 nM T99840 CU3E6Y 67415655 IC50 = 78 nM T99840 CF5O8P 67416617 IC50 = 213 nM T99840 CDW41V 67416619 IC50 = 442 nM T99840 CUNK26 67606457 IC50 = 1290 nM T99840 C0MZW4 67606625 IC50 = 500 nM T99840 CL32WA 67606646 IC50 = 8 nM T99840 C9ZJG3 67606672 IC50 = 5 nM T99840 C8CDK5 67606898 IC50 = 135 nM T99840 CV24MS 67606993 IC50 = 710 nM T99840 C49FSK 67607034 IC50 = 52 nM T99840 CQK9F4 67607104 IC50 = 26 nM T99840 CNB15W 67607112 IC50 = 71 nM T99840 CHV08X 67607304 IC50 = 41 nM T99840 C9K5CH 67607317 IC50 = 85 nM T99840 C7N3OX 67607483 IC50 = 280 nM T99840 C37AUI 67607647 IC50 = 27 nM T99840 CT98SM 67607867 IC50 = 11 nM T99840 CX5P7E 67607972 IC50 = 200 nM T99840 C51DEJ 67608037 IC50 = 770 nM T99840 CYX9E6 67608092 IC50 = 45 nM T99840 CVGQ61 67608205 IC50 = 178 nM T99840 CR05TQ 67608430 IC50 = 260 nM T99840 C6FL8Y 67608513 IC50 = 36 nM T99840 CG2OR6 67608703 IC50 = 850 nM T99840 C7Q0LN 67608774 IC50 = 160 nM T99840 CF3S1G 67608840 IC50 = 15 nM T99840 C3PCZ7 67608997 IC50 = 320 nM T99840 CSR21X 67609024 IC50 = 76 nM T99840 C58NAQ 67609354 IC50 = 260 nM T99840 C7H5FX 67609505 IC50 = 603 nM T99840 CPXI26 67700435 IC50 = 1060 nM T99840 CGA89H 68379817 IC50 = 72 nM T99840 CHY40W 68379998 IC50 = 104 nM T99840 C1B6AK 68380073 IC50 = 73 nM T99840 CPA95O 68380152 IC50 = 252 nM T99840 C95VPL 68380260 IC50 = 101 nM T99840 CLBY90 68380304 IC50 = 6 nM T99840 CSC74R 68380314 IC50 = 128 nM T99840 C07ZLW 68380403 IC50 = 302 nM T99840 C02UKY 68380472 IC50 = 15 nM T99840 CM61LR 68495004 IC50 = 580 nM T99840 C0OPQ6 68495695 IC50 = 130 nM T99840 CXU94C 68624921 IC50 = 300 nM T99840 CH5FN4 69491281 IC50 = 140 nM T99840 CC8QU9 70227534 IC50 = 24 nM T99840 CT71PW 70271003 IC50 = 550 nM T99840 CA27SR 70681184 IC50 = 2070 nM T99840 C23CRI 70681196 IC50 = 1090 nM T99840 CH4Z3G 70681292 IC50 = 110 nM T99840 C1UBD3 70683285 IC50 = 300 nM T99840 CJ4P9D 70683379 IC50 = 110 nM T99840 CEZ21F 70683380 IC50 = 90 nM T99840 CNH04A 70685394 IC50 = 7420 nM T99840 CP6KD8 70685475 IC50 = 50 nM T99840 CBO7F4 70685476 IC50 = 210 nM T99840 CR31EK 70685477 IC50 = 120 nM T99840 CK1G2I 70686452 IC50 = 1.04 nM T99840 C3S8PO 70687527 IC50 = 817 nM T99840 CL8W4C 70687532 IC50 = 160 nM T99840 CR73XZ 70687533 IC50 = 420 nM T99840 C85ORZ 70687534 IC50 = 80 nM T99840 CFO9M4 70687535 IC50 = 80 nM T99840 C6JX3Q 70687593 IC50 = 2600 nM T99840 C3JM6F 70687626 IC50 = 190 nM T99840 CTD2H6 70687627 IC50 = 80 nM T99840 CFQ49O 70687628 IC50 = 160 nM T99840 CF6VM9 70687629 IC50 = 80 nM T99840 C6HN4A 70687630 IC50 = 30 nM T99840 C73WJM 70688498 IC50 > 5000 nM T99840 CIE2O6 70689591 IC50 = 330 nM T99840 CHAV16 70689592 IC50 = 70 nM T99840 CMGO80 70689593 IC50 = 290 nM T99840 CP0O2M 70689684 IC50 > 10000 nM T99840 CNMC10 70689685 IC50 = 400 nM T99840 COB0T1 70689686 IC50 = 60 nM T99840 C1FL0M 70689687 IC50 = 50 nM T99840 C2N1MW 70691706 IC50 = 230 nM T99840 C14ZJR 70691707 IC50 = 430 nM T99840 CV1X9D 70691822 IC50 = 70 nM T99840 CR30DQ 70693785 IC50 = 240 nM T99840 C1RM3T 70693787 IC50 = 30 nM T99840 C52LMB 70693791 IC50 = 1330 nM T99840 C6F3YP 70693884 IC50 = 180 nM T99840 CZX6V9 70693885 IC50 = 50 nM T99840 CS35JI 70693886 IC50 = 640 nM T99840 CSQ1U4 70695560 IC50 = 12 nM T99840 CFB1W2 70695912 IC50 = 20 nM T99840 CX1YS3 70695995 IC50 = 120 nM T99840 CLGU94 70695996 IC50 = 970 nM T99840 CNF49O 70696795 IC50 > 5000 nM T99840 CLA17Z 70696796 IC50 > 5000 nM T99840 CMNO49 71192383 IC50 = 8 nM T99840 CU94LC 71260392 EC50 = 90 nM T99840 CD34HG 71450203 IC50 = 6400 nM T99840 C7SX3I 71450567 IC50 = 11500 nM T99840 CYBE17 71452399 IC50 = 17700 nM T99840 C2EI0Q 71452401 IC50 > 160000 nM T99840 CK85SQ 71452402 IC50 = 7300 nM T99840 C01WUF 71453831 IC50 = 16 nM T99840 CWS9B6 71454178 IC50 = 17700 nM T99840 C7E8LW 71455562 IC50 = 46 nM T99840 CZ0FR2 71455918 IC50 > 40000 nM T99840 CN0G2Y 71457197 IC50 = 100 nM T99840 CHA1Y2 71457710 IC50 = 10000 nM T99840 CO3G6C 71457711 IC50 > 40000 nM T99840 CCW60T 71457712 IC50 = 19800 nM T99840 CNI6L3 71457713 IC50 = 4700 nM T99840 C38SKG 71459162 IC50 = 35 nM T99840 CD5H1K 71459215 IC50 = 48 nM T99840 C2Y7EV 71459621 IC50 = 7600 nM T99840 CG1LN5 71459622 IC50 = 11500 nM T99840 C1ER2C 71459623 IC50 > 80000 nM T99840 CE0L8Q 71459624 IC50 = 27600 nM T99840 CUTC89 71461361 IC50 = 27300 nM T99840 CELP71 71461362 IC50 = 38800 nM T99840 CE32BY 71461363 IC50 = 6700 nM T99840 CBO83G 71461364 IC50 = 47600 nM T99840 CZ9YK5 71462725 IC50 = 11 nM T99840 CRQ6N1 71463084 IC50 = 11300 nM T99840 CK46IV 71463085 IC50 = 5400 nM T99840 C6YD9K 71520616 IC50 = 4.5 nM T99840 C2PEI6 71520617 IC50 = 2.7 nM T99840 CJO7I6 71520701 IC50 = 2.1 nM T99840 CE34VC 71520702 IC50 = 1.4 nM T99840 CCF8I9 71520703 IC50 = 4.7 nM T99840 CD9B7C 71520704 IC50 = 4.3 nM T99840 CD64QG 71520705 IC50 = 1.2 nM T99840 C6S3AU 71520806 IC50 = 1.8 nM T99840 CTX49K 71520807 IC50 = 21 nM T99840 C9GUD6 71520808 IC50 = 1.9 nM T99840 C2N5RD 71520810 IC50 = 280 nM T99840 C8TJK7 71520903 IC50 = 25 nM T99840 CN3CI9 71520904 IC50 = 3.5 nM T99840 C45VZB 71524727 IC50 = 10000 nM T99840 C3Z8EL 71524730 IC50 = 10000 nM T99840 C3TYR5 71524781 IC50 = 10000 nM T99840 CLG84N 71540051 IC50 = 43 nM T99840 CL5I0G 71540052 IC50 = 64 nM T99840 CH5N7C 71540152 IC50 = 53 nM T99840 C8NG0Y 71540153 IC50 = 41 nM T99840 C7XN9A 71552168 IC50 = 0.4 nM T99840 C1V5ZC 71552188 IC50 = 39 nM T99840 C6ES2P 71552253 IC50 = 0.4 nM T99840 C3SH2B 71557331 IC50 = 250 nM T99840 CF24JA 71557332 IC50 = 120 nM T99840 CC47DA 71557333 IC50 = 310 nM T99840 C09VTA 71557334 IC50 = 460 nM T99840 C1HS2T 71557500 IC50 = 260 nM T99840 CE9G0B 71557501 IC50 = 29 nM T99840 CS7JM4 71557502 IC50 = 190 nM T99840 C72SHC 71557504 IC50 = 110 nM T99840 C75RON 71557655 IC50 = 200 nM T99840 CURK41 71557656 IC50 = 510 nM T99840 C62QLB 71557817 IC50 = 290 nM T99840 C38SQK 71574724 IC50 > 30000 nM T99840 C0RY5D 71574725 IC50 > 30000 nM T99840 CLPB03 71574822 IC50 > 30000 nM T99840 COV8K9 71574823 IC50 = 2280 nM T99840 CBE97Z 71574913 IC50 > 30000 nM T99840 CK4YB7 71574914 IC50 = 225 nM T99840 C07NVU 71575007 IC50 = 3.16 nM T99840 CPO3K8 71575103 IC50 = 2.47 nM T99840 C27ADL 71623049 EC50 = 67 nM T99840 C1Q9HS 71680619 EC50 = 22 nM T99840 CH0R3N 71680621 EC50 = 46 nM T99840 CI27WN 71716136 IC50 = 78 nM T99840 C1P4JM 71716463 IC50 = 0.402 nM T99840 CD1AG0 71718313 IC50 > 30000 nM T99840 CZT3I5 71718332 IC50 = 10000 nM T99840 CUZ34P 71746393 IC50 = 43 nM T99840 CA6V3F 71746394 IC50 = 2.1 nM T99840 CD4OV3 71746395 IC50 = 0.33 nM T99840 CSU27O 71746396 IC50 = 1.4 nM T99840 C94KHS 71746397 IC50 = 0.18 nM T99840 CQ1UL5 71746584 IC50 = 0.14 nM T99840 CDEN65 72543942 IC50 > 10000 nM T99840 CR9F6I 72543943 IC50 > 10000 nM T99840 C16ZBK 72543944 IC50 = 1450 nM T99840 CC7T5S 72543945 IC50 = 1530 nM T99840 CXC37J 72543946 IC50 = 1350 nM T99840 CO7JZ1 72543947 IC50 > 10000 nM T99840 CSY96R 72544183 IC50 > 10000 nM T99840 CZQ56P 72544184 IC50 > 10000 nM T99840 CW3BR0 72544185 IC50 = 1110 nM T99840 CFA8B5 72544186 IC50 > 10000 nM T99840 CD8Z0S 72544187 IC50 = 2120 nM T99840 C3YST0 72544408 IC50 = 320 nM T99840 C4XR6N 72544409 IC50 > 10000 nM T99840 C6Z9HC 72544410 IC50 = 2130 nM T99840 COQ63R 72544411 IC50 = 820 nM T99840 C3EJ1X 72544412 IC50 > 10000 nM T99840 CV2BY4 72544413 IC50 = 7000 nM T99840 CFLQ91 72544633 IC50 = 570 nM T99840 C3H5VB 72544634 IC50 > 10000 nM T99840 CX7P3D 72544856 IC50 > 10000 nM T99840 CMLI62 72544858 IC50 = 260 nM T99840 C0UPR3 72545078 IC50 > 10000 nM T99840 C3UE9I 72545079 IC50 = 250 nM T99840 C58EVN 72545080 IC50 = 570 nM T99840 C26ABP 72545081 IC50 = 150 nM T99840 C7QIO8 72545318 IC50 = 20 nM T99840 C3PXJ6 72545565 IC50 = 1290 nM T99840 C8JLR9 72545566 IC50 = 150 nM T99840 C34JIF 72545567 IC50 = 650 nM T99840 CA7Y1S 72547022 IC50 > 10000 nM T99840 CW24CT 72547023 IC50 = 2440 nM T99840 C2NCW7 72547024 IC50 > 10000 nM T99840 C7W9JZ 72547025 IC50 > 10000 nM T99840 C1I6VN 72547026 IC50 = 2100 nM T99840 C0Y6IK 72547282 IC50 = 9400 nM T99840 CK50CR 72547283 IC50 = 2750 nM T99840 CZI51W 72547284 IC50 > 10000 nM T99840 C3PTC5 72547285 IC50 > 10000 nM T99840 CY5DQ1 72547286 IC50 = 720 nM T99840 C5XCD4 72547287 IC50 = 280 nM T99840 C4D6PL 72547528 IC50 = 530 nM T99840 CPSB14 72547529 IC50 = 1830 nM T99840 CY91WF 72547530 IC50 = 1260 nM T99840 C48CJQ 72547531 IC50 = 210 nM T99840 CGTC61 72547532 IC50 = 4060 nM T99840 C81YEF 72547533 IC50 > 10000 nM T99840 CE86LF 73345935 IC50 = 1 nM T99840 CWKT40 73345936 IC50 = 60.9 nM T99840 CAF7D6 73345937 IC50 = 133 nM T99840 CA9NC4 73347460 IC50 = 4.6 nM T99840 CPZ91F 73348985 IC50 = 45 nM T99840 CUJ6D8 73350541 IC50 = 117 nM T99840 CG60TJ 73350542 IC50 = 0.3 nM T99840 C30CPA 73350543 IC50 = 47 nM T99840 CP49WL 73352062 IC50 = 0.22 nM T99840 CJ54XQ 73355022 IC50 = 122 nM T99840 CUQ8P7 73355689 IC50 = 62.6 nM T99840 CHAX61 73356579 IC50 = 662 nM T99840 CQ5EP8 73356580 IC50 = 1.86 nM T99840 CYX9E7 73356581 IC50 = 127 nM T99840 CVD9I2 73356582 IC50 = 9.4 nM T99840 C5C7BQ 73441861 EC50 = 14 nM T99840 CFNG54 73441862 EC50 = 9 nM T99840 CE9S7G 73441910 EC50 = 8 nM T99840 C7RAQ4 74538704 IC50 = 2 nM T99840 CC8X5N 75026445 IC50 = 159 nM T99840 CMG4W9 75026446 IC50 = 34 nM T99840 C3S9XM 75593327 EC50 = 50 nM T99840 C0VR9U 76283428 IC50 = 12 nM T99840 CM0CX5 76283429 IC50 = 13 nM T99840 C20YHA 76283431 IC50 = 228 nM T99840 CE2FS3 76283432 IC50 = 5 nM T99840 CHV72I 76283681 IC50 = 25 nM T99840 CT59ZA 76283684 IC50 = 3 nM T99840 CL76SU 76311131 IC50 = 920 nM T99840 C5GQ4Y 76311132 IC50 = 410 nM T99840 CCY61I 76314929 IC50 = 33 nM T99840 CA90TO 76314930 IC50 = 20 nM T99840 CON91Y 76318326 IC50 = 400 nM T99840 C6LD1Z 76318327 IC50 = 1635 nM T99840 C7HW8O 76318328 IC50 = 311 nM T99840 C78SKI 76318329 IC50 = 135 nM T99840 CPN80M 76318550 IC50 = 1.5 nM T99840 CXJT49 76322016 IC50 = 1498 nM T99840 CKX8R9 76325826 IC50 = 12 nM T99840 C1K4DW 76329211 IC50 = 3400 nM T99840 CXTC05 76329212 IC50 = 530 nM T99840 C1T9YD 76329416 IC50 = 23 nM T99840 C63HQJ 76332863 IC50 = 1270 nM T99840 CE47PB 76333057 IC50 = 1 nM T99840 CM1G0K 76336477 IC50 > 15800 nM T99840 CZK4H7 76336685 IC50 = 180 nM T99840 C0H6RM 88313830 IC50 = 790 nM T99840 CNK3Q7 88875492 IC50 = 86 nM T99840 CQ5VJ6 88875808 IC50 = 87 nM T99840 CF67AV 88875879 IC50 = 63 nM T99840 C7ZV5N 89554314 IC50 = 130 nM T99840 CJSP78 89554316 IC50 = 150 nM T99840 C73HFI 89657800 IC50 = 294 nM T99840 C61XRT 89657803 IC50 = 208 nM T99840 C2UX5Q 89657806 EC50 = 347 nM T99840 C5N4FH 89657810 IC50 = 163 nM T99840 CFJ76Q 89657814 EC50 = 1300 nM T99840 CWRS81 89908079 IC50 = 8 nM T99840 C9VQ2W 90174377 IC50 = 112 nM T99840 C14MXT 90667691 IC50 = 100 nM T99840 C4LWC3 90667692 IC50 = 9800 nM T99840 CPMS46 90667839 IC50 = 60 nM T99840 C3O7HA 90667840 IC50 = 600 nM T99840 C2X1ZG 90667841 IC50 = 3100 nM T99840 CAK3F9 90667842 IC50 = 760 nM T99840 C69TWF 90667843 IC50 = 8400 nM T99840 C89UCI 90667844 IC50 = 95 nM T99840 CM0Z9Y 90667845 IC50 = 520 nM T99840 C6WYN1 90667846 IC50 = 260 nM T99840 CER7B8 90667847 IC50 = 1000 nM T99840 CJK62Z 90667848 IC50 = 780 nM T99840 CK7SA3 90667849 IC50 = 1600 nM T99840 CVZ65U 90667850 IC50 = 4600 nM T99840 CYPQ69 90667851 IC50 = 860 nM T99840 CZ7B4N 90667852 IC50 = 590 nM T99840 C8W2RG 90667853 IC50 = 1300 nM T99840 C26GUK 90667854 IC50 = 220 nM T99840 CFXY12 90667855 IC50 = 200 nM T99840 C62PWT 90667856 IC50 = 3000 nM T99840 C8ANE3 90667857 IC50 = 360 nM T99840 C0PGO5 90667858 IC50 = 230 nM T99840 C92COG 90667859 IC50 = 470 nM T99840 C9TW7Y 90667860 IC50 = 47 nM T99840 C7OPI4 90667861 IC50 = 450 nM T99840 CQTM43 90667862 IC50 = 560 nM T99840 CIAD34 90667863 IC50 = 84 nM T99840 CNU18A 90667864 IC50 = 2500 nM T99840 CWEF89 90667865 IC50 = 340 nM T99840 CU7K8Z 90667866 IC50 = 220 nM T99840 CZI63D 91755037 EC50 = 14 nM T99840 CSK6Z1 91844707 IC50 = 14 nM T99840 CK6O3J 92042908 IC50 = 6 nM T99840 CJ23FH 95180362 IC50 = 150 nM T99840 CK02NB 101593793 IC50 = 6250 nM T99840 CGK2W6 118003167 IC50 = 52 nM T99840 CSN6A7 118003183 IC50 = 9 nM T99840 CL0P4E 118003318 IC50 = 389 nM T99840 C2E6WF 118049905 IC50 = 58.5 nM T99840 CDBI46 118049974 EC50 = 105 nM T99840 CW54AG 118049998 IC50 = 30.5 nM T99840 CV3EL4 118050047 IC50 = 25.6 nM T99840 CJ9L0H 118050068 IC50 = 25.4 nM T99840 CA10PR 118050100 IC50 = 72.4 nM T99840 CEQV79 118050174 IC50 = 20.8 nM T99840 CRUP56 118051801 EC50 = 39 nM T99840 C6MQU8 118051925 EC50 = 101 nM T99840 C1SH7T 118054978 IC50 = 54.3 nM T99840 C8L5NJ 118055002 EC50 = 25 nM T99840 C2U9FP 118055004 IC50 = 54.8 nM T99840 CH08WQ 118055008 IC50 = 11.9 nM T99840 CP0CN6 118055017 IC50 = 90 nM T99840 C3PJN1 118055019 IC50 = 56 nM T99840 CT2XV3 118238206 EC50 = 16 nM T99840 CTJN74 118246000 EC50 = 49 nM T99840 CR94TZ 118246257 EC50 = 71 nM T99840 CQH93R 118389830 IC50 = 129 nM T99840 C2E3HO 118389852 IC50 = 13 nM T99840 C50EMF 118389864 IC50 = 4.9 nM T99840 C42MCT 118389887 IC50 = 181 nM T99840 CNC75S 118389896 IC50 = 5.1 nM T99840 C76YWL 118389909 IC50 = 6 nM T99840 CS75HY 118389912 IC50 = 52 nM T99840 CBIR89 118389918 IC50 = 4.9 nM T99840 CN4F6I 118389934 IC50 = 5.6 nM T99840 C24EQN 118389941 IC50 = 801 nM T99840 C70EHC 118389944 IC50 = 53 nM T99840 CT8NU9 118390140 IC50 = 63 nM T99840 CGZP63 118390142 IC50 = 322 nM T99840 C46CPT 118403551 IC50 = 30 nM T99840 CM2NH5 118478848 IC50 = 250.7 nM T99840 CAS3Q9 118717940 IC50 = 25.12 nM T99840 C3GU9R 118717942 IC50 = 1584.89 nM T99840 C6PGA5 118717943 IC50 = 39.81 nM T99840 C7MT5V 118717944 IC50 = 19.95 nM T99840 CX0E4Z 118717945 IC50 = 39.81 nM T99840 CXBW96 118717946 IC50 = 12.59 nM T99840 C5PY4C 118717947 IC50 = 10 nM T99840 CZQB45 118717948 IC50 = 10 nM T99840 C8GVY4 118717949 IC50 = 15848.93 nM T99840 C5N3XM 118717950 IC50 = 19.95 nM T99840 CM1W4V 118717951 IC50 = 316.23 nM T99840 C8ZD5R 118717953 IC50 = 15.85 nM T99840 C2GD7Q 118717957 IC50 = 39.81 nM T99840 CATJ63 118717964 IC50 = 10 nM T99840 CQ42VG 118717965 IC50 = 31.62 nM T99840 C5FS2H 118717970 IC50 = 63.1 nM T99840 C8G0VO 118717971 IC50 = 12.59 nM T99840 C8A2MI 118717972 IC50 = 10000 nM T99840 CAI6Y5 118717973 IC50 = 63.1 nM T99840 CYOM60 118717977 IC50 = 158.49 nM T99840 CT2L5C 118717979 IC50 = 12.59 nM T99840 CZW41X 118717980 IC50 = 19.95 nM T99840 CB3Y8R 118717981 IC50 = 100 nM T99840 C6DLS9 118717982 IC50 = 39.81 nM T99840 C92TQH 118717986 IC50 = 1258.93 nM T99840 CT6MH3 118717989 IC50 = 50.12 nM T99840 CC07RJ 118719411 IC50 = 22 nM T99840 C0S1FZ 118719628 IC50 = 140 nM T99840 C2TWM9 118719629 IC50 = 58 nM T99840 CY0K7Z 118719630 IC50 = 340 nM T99840 CGK38C 118719631 IC50 = 670 nM T99840 CSP43R 118726362 IC50 = 234 nM T99840 CD2E8S 118726363 IC50 = 42 nM T99840 C6WB1O 118726364 IC50 = 19 nM T99840 C87UJQ 118726365 IC50 = 207 nM T99840 CD0CG9 118726366 IC50 = 128 nM T99840 C1O6GD 118726367 IC50 = 96 nM T99840 CX5G2H 118726368 IC50 = 44 nM T99840 CLMU64 118726369 IC50 = 38 nM T99840 CDX1G4 118726370 IC50 = 17 nM T99840 C21WVF 118726371 IC50 = 92 nM T99840 CGC48T 118726372 IC50 = 170 nM T99840 CQB7L8 118726373 IC50 = 361 nM T99840 CFJ1O9 118726374 IC50 = 418 nM T99840 C1KCQ3 118726375 IC50 = 142 nM T99840 CYPG84 118726376 IC50 = 605 nM T99840 CJ6OE8 118726377 IC50 = 22 nM T99840 CLO50Q 118726378 IC50 = 35 nM T99840 CR9NH6 122178430 IC50 = 20 nM T99840 CQ10JD 122178431 IC50 = 85 nM T99840 C80QLF 122186844 IC50 = 5310 nM T99840 CF47TW 122186845 IC50 = 70 nM T99840 CQM3Z7 122186846 IC50 = 110 nM T99840 CKD2V7 122186847 IC50 = 36 nM T99840 C6UGI9 122186848 IC50 = 350 nM T99840 C3MZN1 122186849 IC50 = 310 nM T99840 CE5C9J 122186850 IC50 = 170 nM T99840 C4Y9AM 122186851 IC50 = 62 nM T99840 CE7LZ2 122186852 IC50 = 10000 nM T99840 CS20UJ 122186853 IC50 = 270 nM T99840 C59JBF 122187726 IC50 = 880 nM T99840 CC7W9L 122187727 IC50 = 40 nM T99840 C2N0KO 122187728 IC50 = 240 nM T99840 CRUK02 122187729 IC50 = 70 nM T99840 C7BF8W 122187730 IC50 = 70 nM T99840 C3DX2S 122187798 IC50 = 56 nM T99840 C9VFM5 122187799 IC50 = 11 nM T99840 CR42XN 122187800 IC50 = 210 nM T99840 C4XCP1 122187801 IC50 = 58 nM T99840 CCU2N7 122187802 IC50 = 13 nM T99840 CT2ZJ6 122187803 IC50 = 1490 nM T99840 CGQ8V9 122187804 IC50 = 260 nM T99840 C5W6XS 124351898 EC50 = 40000 nM T99840 CM25EQ 124660563 IC50 = 0.41 nM T99840 CO4Z8M 127025082 IC50 = 1200 nM T99840 CX47HA 127025378 IC50 = 180 nM T99840 CS1CE6 127025655 IC50 = 140 nM T99840 CK2WV4 127028395 IC50 = 35 nM T99840 CN4W1K 127028397 IC50 = 140 nM T99840 CKI9F8 127028409 IC50 = 20 nM T99840 CK79WY 127028410 IC50 = 1800 nM T99840 CD52OH 127028411 IC50 = 50 nM T99840 CP56WJ 127028412 IC50 = 80 nM T99840 C8A4GZ 127028413 IC50 = 120 nM T99840 CZ72JM 127028414 IC50 = 300 nM T99840 C5FZ7T 127028415 IC50 = 1100 nM T99840 CGR4U3 127028416 IC50 = 380 nM T99840 CH4M9N 127028417 IC50 = 1000 nM T99840 C1R8JC 127028418 IC50 = 50 nM T99840 C8W7QS 127028419 IC50 = 190 nM T99840 C1CWF9 127028424 IC50 = 460 nM T99840 CQM96C 127028425 IC50 = 820 nM T99840 CU1CN2 127028426 IC50 = 100 nM T99840 C9R3XB 127028427 IC50 = 200 nM T99840 CZ59BG 127029070 IC50 = 5 nM T99840 C3N8RT 127029071 IC50 = 21 nM T99840 CZBU47 127029072 IC50 = 36 nM T99840 CPY1N6 127029350 IC50 = 56 nM T99840 C3IXT1 127030015 IC50 = 95000 nM T99840 CV10UT 127030331 IC50 = 580 nM T99840 C28VXD 127030332 IC50 = 360 nM T99840 C23GEY 127046417 IC50 = 26000 nM T99840 CY5W9Z 127047958 IC50 > 75000 nM T99840 CCQ7Y5 127053276 IC50 = 135000 nM T99840 CL6O9Z 127053277 IC50 = 85000 nM T99840 C32JOQ 135858933 IC50 = 72 nM T99840 C23LZV 135869398 IC50 = 411 nM T99840 CS56QT 135869399 IC50 = 220 nM T99840 CW6RJ7 135869400 IC50 = 287 nM T99840 CE13WD 135869401 IC50 = 250 nM T99840 C3LP9O 135869402 IC50 = 163 nM T99840 C51QDS 135869403 IC50 = 111 nM T99840 C3ANW7 135869404 IC50 = 88 nM T99840 CU42ZL 135869405 IC50 = 258 nM T99840 C81QEC 135869406 IC50 = 287 nM T99840 C0B6PF 135869407 IC50 = 218 nM T99840 CN4KG1 135869408 IC50 = 301 nM T99840 CW7Q3G 135878222 IC50 = 85 nM T99840 C72FKJ 135878229 IC50 = 92 nM T99840 CB6EV1 135878230 IC50 = 63 nM T99840 CB9M6Z 135878231 IC50 = 158 nM T99840 C19SRN 135878240 IC50 = 91 nM T99840 CTW0K3 135899156 IC50 = 0.65 nM T99840 CBX90O 135910326 IC50 = 3890 nM T99840 C5EC2O 135910327 IC50 = 660 nM T99840 C4AI7G 136030608 IC50 = 4280 nM T99840 C2HP1X 136030609 IC50 = 6740 nM T99840 CCZO92 136030610 IC50 = 3740 nM T99840 CCQ51T 136030757 IC50 = 4870 nM T99840 C0RU6A 136053698 IC50 = 180 nM T99840 C8AZJ9 136069091 IC50 = 20000 nM T99840 C1U8TM 136160538 IC50 = 340 nM T99840 C9QF0C 136199922 IC50 = 171 nM T99840 CDE9Z1 136224008 IC50 = 0.56 nM T99840 CL74HF 136229224 IC50 = 72 nM T99840 C0XLT5 136264485 IC50 = 1 nM T99840 CW83TZ 136626667 IC50 = 36 nM T99840 CPK9S5 136626671 IC50 = 107 nM T99840 C3NG2Q 136626673 IC50 = 25 nM T99840 CZPV15 136626674 IC50 = 117 nM T99840 C2OSQ1 136627167 IC50 = 3981 nM T99840 C0UP1A 137174951 IC50 = 40 nM T99840 CJC95O 138319684 IC50 = 40 nM T99840 CQE13R 138678573 EC50 = 14 nM T99840 CQ5E0B 138678593 EC50 = 111 nM T99840 C8QH0O 138678605 EC50 = 34 nM T99840 C7H9KZ 138678606 EC50 = 19 nM T99840 C1FZ7S 138678620 EC50 = 35 nM T99840 CLHK06 138678794 EC50 = 36 nM T99840 C2AOQ9 139415485 EC50 = 5 nM T99840 CCT8G2 139415505 EC50 = 8 nM T99840 C3K2ZI 139415517 EC50 = 13 nM T99840 C75SJT 139415533 EC50 = 15 nM T99840 CH62KO 139415536 EC50 = 8 nM T99840 CDM5L3 139415543 EC50 = 33 nM T99840 C0M5IB 139415544 EC50 = 7 nM T99840 C6VF5T 139430688 EC50 = 30 nM T99840 CT1L7K 142606858 IC50 = 14 nM T99840 C0RAK9 142606862 IC50 = 8 nM T99840 CQL72N 142606863 IC50 = 25 nM T99840 CZ4W2M 142606877 IC50 = 49 nM T99840 C65IWN 142606880 IC50 = 27 nM T99840 CG23NY 142606884 IC50 = 16 nM T99840 C1GD8S 142606886 IC50 = 44 nM T99840 CZW98E 142606887 IC50 = 15 nM T99840 C4YPQ7 142606891 IC50 = 23 nM T99840 CO70HU 142606893 IC50 = 31 nM T99840 CU6SN1 142606894 IC50 = 15 nM T99840 C94CBQ 142606895 IC50 = 14 nM T99840 CXV31J 142606896 IC50 = 26 nM T99840 C05MIP 142607769 IC50 = 120 nM T99840 C1LR5J 142607770 IC50 = 1200 nM T99840 C3TMR0 142607778 IC50 = 90 nM T99840 CMFQ84 142607794 IC50 = 2770 nM T99840 C0VR9Y 142607800 IC50 = 350 nM T99840 CE1B9H 142607803 IC50 = 3400 nM T99840 C34GVD 142607804 IC50 = 200 nM T99840 CZYG08 142607806 IC50 = 30 nM T99840 C7MUQ2 142607808 IC50 > 30000 nM T99840 C8TM1A 142607812 IC50 = 70 nM T99840 CO08KN 142607816 IC50 = 40 nM T99840 CPHZ53 142607820 IC50 = 194 nM T99840 CR01WI 142607828 IC50 > 30000 nM T99840 CDZ91R 142607841 IC50 = 60 nM T99840 CN09SF 142607846 IC50 = 730 nM T99840 CL3D6V 142607847 IC50 = 1390 nM T99840 CF79IB 142607849 IC50 = 4570 nM T99840 CA8TY4 142607851 IC50 = 200 nM T99840 C5A1MS 142607854 IC50 = 3130 nM T99840 CY6FI1 142607870 IC50 = 680 nM T99840 CBX8T3 142607871 IC50 = 750 nM T99840 C3B0JS 142607879 IC50 = 670 nM T99840 CBD2L5 142607880 IC50 = 430 nM T99840 CU39BH 142607882 IC50 = 50 nM T99840 C7KTU5 142607897 IC50 = 740 nM T99840 C73HXD 142607900 IC50 = 380 nM T99840 CZ91AK 145955876 IC50 = 21700 nM T99840 CS6Z9D 145961223 IC50 = 180 nM T99840 CHR50A 145961243 IC50 = 60 nM T99840 CQ0YK2 145961280 IC50 = 500 nM T99840 C6ID3H 145961522 IC50 = 2200 nM T99840 CSB5U8 145961774 IC50 = 60 nM T99840 CWI9B1 145961933 IC50 = 20 nM T99840 CWB80D 145962590 IC50 = 40 nM T99840 CJ5A6Q 145962645 IC50 = 950 nM T99840 C4H9TL 145963152 IC50 = 160 nM T99840 CE7UM2 145963197 IC50 = 70 nM T99840 CCRH49 145963599 IC50 = 9 nM T99840 CIQ30C 145963822 IC50 > 50000 nM T99840 C5E3FO 145964932 IC50 = 690 nM T99840 CC9QL4 145966531 IC50 = 1800 nM T99840 CQV46Y 145970305 IC50 = 17 nM T99840 CDTU34 145970496 IC50 > 10000 nM T99840 CKH7U4 145972721 IC50 = 1300 nM T99840 CJ0US7 145973873 IC50 = 7100 nM T99840 C2SQV7 145974463 IC50 = 390 nM T99840 C0DWZ2 145976055 IC50 = 9800 nM T99840 CVF1G3 145977207 IC50 = 5800 nM T99840 CFZA28 145977593 IC50 > 50000 nM T99840 CEX8V9 145978454 IC50 = 8700 nM T99840 C4HQO0 145978536 IC50 = 2300 nM T99840 CO5RK9 145988561 EC50 = 14 nM T99840 CLO3W7 145992890 EC50 = 8 nM T99840 C73LTZ 146306592 EC50 = 0.013 nM T99840 CD6KR9 146306602 EC50 = 0.0103 nM T99840 C7O4XE 146306604 EC50 = 0.0114 nM T99840 CR9V2L 146306617 EC50 = 0.0117 nM T99840 CT3H9B 146306631 EC50 = 0.0059 nM T99840 CO69MS 155164669 IC50 = 39 nM T99840 CQ1EW0 155510983 EC50 = 10 nM T99840 CT4LJ1 155512934 IC50 = 41 nM T99840 C24AKY 155513525 IC50 = 175 nM T99840 C2DSZ8 155513622 EC50 = 6 nM T99840 COQX09 155515761 IC50 > 1000 nM T99840 C94IPH 155517286 IC50 = 110 nM T99840 CVAI54 155517459 EC50 = 20 nM T99840 CKZ7Y8 155518783 IC50 = 45 nM T99840 C5QGD4 155519995 IC50 = 98 nM T99840 C1AZB0 155520838 IC50 = 475 nM T99840 CIC5L7 155521256 IC50 = 603 nM T99840 C3KSY8 155522962 EC50 = 45 nM T99840 CRH81M 155523684 IC50 = 179 nM T99840 CFA5X1 155524819 IC50 = 362 nM T99840 CQXZ91 155525880 IC50 = 114 nM T99840 CAM48S 155526231 EC50 = 0.0092 nM T99840 C69CBF 155526641 IC50 = 18 nM T99840 CD5QT6 155526690 IC50 > 1000 nM T99840 C50HCX 155526887 IC50 = 216 nM T99840 CC1O5K 155530531 IC50 = 49 nM T99840 CUW4Z9 155530939 IC50 = 394 nM T99840 CSU48Z 155531407 IC50 = 148 nM T99840 CFL61W 155532250 IC50 = 19 nM T99840 CE8Y0F 155532723 IC50 = 112 nM T99840 C18XWC 155533276 IC50 = 225 nM T99840 C0PD6N 155533341 IC50 = 219 nM T99840 CM6HK5 155533472 IC50 = 55 nM T99840 C2QHX4 155534806 IC50 = 15 nM T99840 CB63DW 155539872 IC50 = 771 nM T99840 CXIS50 155540564 IC50 = 280 nM T99840 C8AJU4 155540955 IC50 > 1000 nM T99840 C4RUM6 155542247 IC50 = 31 nM T99840 C6IVD9 155542803 IC50 = 23 nM T99840 C0TDZ4 155544576 IC50 = 270 nM T99840 CEY5H1 155544970 IC50 = 87 nM T99840 C0F3HL 155546703 IC50 = 4000 nM T99840 CG50LE 155547624 IC50 > 1000 nM T99840 CA5ID2 155547685 IC50 = 110 nM T99840 CV9LR8 155547786 IC50 = 39 nM T99840 C65HFR 155547882 EC50 = 0.0139 nM T99840 CB9V6O 155548351 EC50 = 21 nM T99840 C27AGI 155549080 EC50 = 6 nM T99840 C9H8MJ 155549445 IC50 = 26 nM T99840 CXQR20 155550079 IC50 = 195 nM T99840 CS5GJ8 155550249 IC50 = 67 nM T99840 C02QZK 155551379 IC50 = 62 nM T99840 CTP2Z9 155551650 IC50 = 36 nM T99840 CNBK91 155552409 IC50 = 32 nM T99840 C9IOT0 155553367 IC50 > 1000 nM T99840 C1GI7C 155554967 IC50 = 66 nM T99840 C4SGF5 155556571 EC50 = 41 nM T99840 C3HMY5 155557465 IC50 = 66 nM T99840 C1SVN7 155558409 IC50 = 41 nM T99840 C0TK7L 155558815 IC50 = 289 nM T99840 CVP1I3 155559282 IC50 = 85 nM T99840 C56CPG 155559540 IC50 = 17 nM T99840 CY05DH 155560260 IC50 = 92 nM T99840 CI5JV9 155560962 IC50 = 94 nM T99840 CV3RC0 155561296 IC50 > 1000 nM T99840 C8NA0K 155562228 IC50 = 347 nM T99840 CR7TI5 155562738 IC50 = 229 nM T99840 C1XZM9 155563081 IC50 = 110 nM T99840 C2H5JE 155565668 IC50 > 1000 nM T99840 CH39OK 155565786 IC50 = 766 nM T99840 CT4GP1 155566638 IC50 = 22 nM T99840 C0CRB1 155567585 IC50 = 121 nM T99840 CM4XS2 155567732 EC50 = 0.0064 nM T99840 C2BDR8 155568466 IC50 = 59 nM T99840 CGWF78 155568726 IC50 = 272 nM T99840 CKYJ21 76283430 IC50 = 6 nM T99840 CIJ3N0 76283682 IC50 = 23.3 nM T99840 D00DFR 11809004 IC50 = 1100 nM T99840 D03AMR 9849669 IC50 = 200 nM T99840 D04TWU 15071517 IC50 = 6900 nM T99840 D0B5FC 447912 EC50 = 3600 nM T99840 D0I8BA 16037828 IC50 = 1000 nM T99840 D0K8LN 44400752 IC50 = 461 nM T99840 D0M2LV 44413811 IC50 = 4900 nM T99840 D0Q6ZQ 53308121 IC50 = 5.3 nM T55948 D05EAM 4735 IC50 = 9500 nM T55948 D07HOB 60838 IC50 = 74600 nM T55948 D0AZ3C 5291 IC50 = 25500 nM T55948 D0K0OZ 5702160 IC50 = 10700 nM T55948 D0K7WK 4595 IC50 = 17400 nM T55948 D0R3JB 4212 IC50 = 60500 nM T55948 D0T6XX 4679 IC50 = 137000 nM T55948 D0V4GY 9552079 IC50 = 410 nM T55948 D0V7CF 5362440 IC50 > 500000 nM T55948 D0ZU9R 392622 IC50 > 300000 nM T55948 D0QQ1J 2406 IC50 = 5500 nM T55948 COC04T 3520 IC50 = 2200000 nM T55948 CP4RM6 4486 IC50 = 146000 nM T55948 C0YU1V 16157 IC50 = 99800 nM T55948 C32CWP 409364 IC50 = 4600 nM T55948 C49RWG 1549311 IC50 = 27800 nM T55948 C4ZUJ5 2757788 IC50 = 2800 nM T55948 CNJ03F 10374840 IC50 = 7600 nM T55948 CVT03F 11265456 IC50 = 1500 nM T55948 CX9Q2G 12420538 IC50 = 4800 nM T55948 C3M1FN 15662596 IC50 = 2200 nM T55948 C4ZD6T 24801038 IC50 = 452500 nM T49898 D00FGR 3599 IC50 > 1000000 nM T49898 D01PZD 5329098 IC50 > 10000 nM T49898 D05SBO 46220502 IC50 > 1000 nM T49898 D08IBS 190 IC50 = 200000 nM T49898 D0G6QF 3081361 IC50 > 10000 nM T49898 D0K8KX 5280343 IC50 = 450 nM T49898 D00UZR 5330286 IC50 > 10000 nM T49898 D03LWG 53235510 IC50 > 10000 nM T49898 D05ADP 160355 IC50 = 330 nM T49898 D06WHY 16747683 IC50 = 62 nM T49898 D08MXP 44631912 IC50 >= 100000 nM T49898 D08UUL 46700756 IC50 > 10000 nM T49898 D0A5MC 11712649 IC50 > 100000 nM T49898 D0CY1B 6420138 Ki > 10000 nM T49898 D0DX4J 67409219 IC50 < 100 nM T49898 D0E3TC 44259 IC50 = 18 nM T49898 D0LF1U 5287969 IC50 = 30 nM T49898 D0M9QZ 11485656 IC50 = 9800 nM T49898 D0P0KN 16739650 IC50 = 3 nM T49898 D0P6DJ 151194 IC50 > 10000 nM T49898 D0S5RC 3025986 Ki = 480 nM T49898 D0WS1V 448991 IC50 = 20000 nM T49898 D00PWQ 3820 IC50 = 400 nM T49898 D07DUX 73353575 IC50 = 50 nM T49898 D0YK9D 9956119 IC50 = 8800 nM T49898 D00BPA 4592 IC50 = 4600 nM T49898 D02YAQ 6603857 IC50 > 8000 nM T49898 D04FHB 6918852 Ki = 2 nM T49898 D09HEV 6539952 IC50 > 20000 nM T49898 D0A9KI 9863367 IC50 > 100 nM T49898 D0D3PX 46926350 IC50 = 3 nM T49898 D0Q7HO 4705 IC50 = 100000 nM T49898 D0U2TQ 644215 IC50 < 5.2 nM T49898 CGAN35 2856 IC50 = 220000 nM T49898 CPZ3I6 3543 IC50 = 52 nM T49898 CHR3Z9 5097 IC50 = 650 nM T49898 C97TNH 10177 IC50 = 10000 nM T49898 C2J0PB 15048 IC50 = 320000 nM T49898 CZJ8U9 30976 IC50 > 100000 nM T49898 C9BIN1 62389 IC50 = 200000 nM T49898 CM1L0U 94904 IC50 > 1000000 nM T49898 CUM2L9 145989 IC50 = 70000 nM T49898 C6Y9CV 151193 IC50 > 10000 nM T49898 C28CSW 158883 IC50 = 214 nM T49898 CR9TJ7 223167 IC50 = 830 nM T49898 CZU0Q6 225611 IC50 = 40000 nM T49898 CA9FO7 245913 IC50 = 2530 nM T49898 CP9Z5G 258725 IC50 = 4900 nM T49898 CMGI79 284815 IC50 = 910 nM T49898 CLW30H 314123 IC50 = 1600 nM T49898 CV3XI1 354479 IC50 > 10000 nM T49898 CY26DN 369402 IC50 = 3300 nM T49898 C8QL0B 383785 IC50 = 600 nM T49898 CY3F2L 383786 IC50 = 1400 nM T49898 C35EWT 383787 IC50 = 1300 nM T49898 CX3A6O 384146 IC50 = 1300 nM T49898 C09JHV 385068 IC50 = 900 nM T49898 C9YCZ3 385069 IC50 = 2000 nM T49898 CUYD71 385070 IC50 = 1600 nM T49898 C06EVW 395169 IC50 = 40000 nM T49898 CDUC10 395170 IC50 = 3000 nM T49898 CUL7P6 395804 IC50 = 300 nM T49898 CG0DM8 395805 IC50 = 200 nM T49898 CZX1J4 396079 IC50 = 400 nM T49898 C0RYZ9 396080 IC50 = 430000 nM T49898 CL0G3P 396081 IC50 = 4300 nM T49898 C3HAR9 396411 IC50 = 250000 nM T49898 C7EN1O 396412 IC50 = 280 nM T49898 CC70DS 396571 IC50 = 240 nM T49898 C0AZN2 396572 IC50 = 2500 nM T49898 CAE9J0 397216 IC50 = 24 nM T49898 CWIQ59 397718 IC50 = 3000 nM T49898 CWSU67 397719 IC50 = 3800 nM T49898 CU1TA8 398149 IC50 > 100000 nM T49898 CH20NR 403176 IC50 = 5 nM T49898 CJV8K2 421101 IC50 = 3230 nM T49898 C4MNG8 445840 IC50 = 122 nM T49898 C9E4FI 447622 IC50 = 2770 nM T49898 CB9F1O 447961 Ki = 80 nM T49898 C6A3LY 447962 Ki = 2520 nM T49898 C1ZG2U 449087 IC50 = 279 nM T49898 C1EB0M 461195 IC50 = 150 nM T49898 CC31FE 512549 IC50 = 160 nM T49898 C2ZN0H 512561 IC50 = 260 nM T49898 C0YIB2 512562 IC50 = 12 nM T49898 C4WFP1 1587957 IC50 > 200000 nM T49898 C1X3LF 2059510 IC50 = 29400 nM T49898 CHC5I0 2971839 IC50 > 10000 nM T49898 CK27QG 3001650 IC50 = 70000 nM T49898 C4ELP8 3160258 IC50 = 3000 nM T49898 C4CA5U 3323623 IC50 = 330 nM T49898 CHGS79 3551941 IC50 = 780 nM T49898 C7RMT3 3960961 IC50 = 200000 nM T49898 C4ZT3K 4155347 IC50 = 100 nM T49898 CR9LG3 4369432 IC50 = 111400 nM T49898 CTXC93 4369433 IC50 = 5000 nM T49898 CN95RS 4477128 IC50 = 2900 nM T49898 CAD5G8 4477129 IC50 = 56 nM T49898 C7NTG0 4477130 IC50 = 19 nM T49898 C0WHD7 4477131 IC50 = 3800 nM T49898 CK3XT1 4477132 IC50 = 2500 nM T49898 CN7MT6 4750207 IC50 > 10000 nM T49898 CS69YO 5032965 IC50 = 2500 nM T49898 CUNA75 5247677 IC50 = 4000000 nM T49898 CHK2V0 5289411 IC50 = 70 nM T49898 CF3Y6G 5327828 IC50 = 5800 nM T49898 CY1Z9E 5327829 IC50 > 1000 nM T49898 CI51CH 5327830 IC50 = 4300 nM T49898 CUAW78 5327831 IC50 = 3000 nM T49898 CC9US2 5327832 IC50 = 57000 nM T49898 CVGK98 5327833 IC50 > 1000 nM T49898 CGWP86 5327834 IC50 = 350 nM T49898 C10RVD 5327835 IC50 = 7400 nM T49898 CD6B2A 5327836 IC50 = 16000 nM T49898 CY1O6K 5327837 IC50 = 3100 nM T49898 C1K8CJ 5327838 IC50 = 5000 nM T49898 CP15JO 5327839 IC50 = 2800 nM T49898 CWT9S8 5327840 IC50 = 200 nM T49898 C5EWD2 5327841 IC50 > 100000 nM T49898 C67JVQ 5327843 IC50 > 100000 nM T49898 CY23QP 5327844 IC50 = 680 nM T49898 CN1X4Z 5327845 IC50 > 100000 nM T49898 C6TGI1 5327846 IC50 = 4500 nM T49898 CB90GI 5327848 IC50 = 9000 nM T49898 CMVG29 5329578 IC50 = 18000 nM T49898 CZG0R9 5329598 IC50 = 63000 nM T49898 CCK8Q5 5329599 IC50 = 5300 nM T49898 CFB24A 5329600 IC50 = 800 nM T49898 CMTY12 5329601 IC50 = 230 nM T49898 CS3CM2 5329602 IC50 = 220 nM T49898 CFQ5N9 5329603 IC50 = 5 nM T49898 C8C3VG 5329674 IC50 = 80 nM T49898 CM9V8E 5329715 IC50 = 130 nM T49898 C4V5QX 5330356 IC50 > 360 nM T49898 CZ3LK2 5330387 IC50 > 10000 nM T49898 CW2MT7 5330397 IC50 = 2400 nM T49898 CH7XF6 5330398 IC50 > 10000 nM T49898 C9ACY8 5330399 IC50 > 10000 nM T49898 CR1CV4 5330401 IC50 > 10000 nM T49898 CSD47J 5330402 IC50 > 10000 nM T49898 C58VWF 5330403 IC50 = 500 nM T49898 CXP8M2 5330404 IC50 = 2220 nM T49898 CGE78Y 5330405 IC50 > 10000 nM T49898 C7E4HZ 5330406 IC50 = 8080 nM T49898 CA7U4J 5330407 IC50 > 10000 nM T49898 C5TGL0 5330583 IC50 = 120 nM T49898 C4J3FI 5331106 IC50 = 1400 nM T49898 CNS20F 5331110 IC50 = 3000 nM T49898 C6W0MJ 5331111 IC50 = 6200 nM T49898 CY91BJ 5331113 IC50 = 6400 nM T49898 CLS0C3 5331114 IC50 = 1000 nM T49898 CXF1P6 5331116 IC50 = 43000 nM T49898 CTNI84 5331118 IC50 = 23000 nM T49898 C1AV7M 5331119 IC50 = 2300 nM T49898 C5KP0C 5331121 IC50 = 20000 nM T49898 C9OW4Y 5331123 IC50 = 70000 nM T49898 CU6V3J 5331124 IC50 = 60000 nM T49898 CS4V6F 5331125 IC50 = 35000 nM T49898 CXK05J 5331126 IC50 = 470000 nM T49898 C2BPX5 5331127 IC50 = 80000 nM T49898 C82ITE 5331130 IC50 = 150000 nM T49898 CB0PR6 5331131 IC50 = 1000000 nM T49898 CPQV76 5353678 IC50 > 100000 nM T49898 CZU0A4 5479542 IC50 > 10000 nM T49898 CRN4I2 6397536 IC50 = 400000 nM T49898 CCRM28 6538898 IC50 = 110 nM T49898 C0O8DH 6538899 IC50 = 600 nM T49898 CW9S3K 6538900 IC50 = 60 nM T49898 C5Y7MX 6538901 IC50 = 9 nM T49898 CZH30S 6538902 IC50 = 800 nM T49898 C8O4ZA 6538904 IC50 = 150000 nM T49898 C1KHR3 6538905 IC50 = 18000 nM T49898 C0VLD2 6538906 IC50 = 11000 nM T49898 C36NRA 6538907 IC50 = 8000 nM T49898 C34REF 6538908 IC50 = 75000 nM T49898 COS29U 6538909 IC50 = 90000 nM T49898 C50PWH 6538910 IC50 = 100000 nM T49898 CU17AZ 6538911 IC50 = 470000 nM T49898 CMV28P 6538912 IC50 = 150000 nM T49898 C7ZBQ5 6538913 IC50 = 110000 nM T49898 CNR9G3 6538914 IC50 = 2100 nM T49898 CZ36MO 6538915 IC50 = 650 nM T49898 C6IV4B 6538916 IC50 = 2500 nM T49898 CXU3H2 6538917 IC50 = 6500 nM T49898 CE1QL2 6538918 IC50 = 2500 nM T49898 C6F5WG 6538919 IC50 = 4300 nM T49898 CL4Z8I 6538920 IC50 = 1000 nM T49898 C7DT1S 6538921 IC50 = 7300 nM T49898 CGH45F 6538922 IC50 = 2700 nM T49898 CJGK38 6538923 IC50 = 900 nM T49898 CMN3A9 6538924 IC50 = 850 nM T49898 CXC4R3 6538925 IC50 = 1000 nM T49898 C5K8QG 6538926 IC50 = 450 nM T49898 CNDE01 6538927 IC50 = 42000 nM T49898 C4VZ3Y 6538928 IC50 = 40000 nM T49898 C5N3IH 6538929 IC50 = 700 nM T49898 CID0S2 6538930 IC50 = 200000 nM T49898 C7JC5M 6538932 IC50 = 230 nM T49898 CUH4Y3 6538933 IC50 = 180 nM T49898 CT7VL8 6538934 IC50 = 200 nM T49898 C1LI8N 6538935 IC50 = 200 nM T49898 CGH31W 6538936 IC50 = 350 nM T49898 CL98HG 6538937 IC50 = 500 nM T49898 CB1Y5Z 6538938 IC50 = 500 nM T49898 CPO71U 6538939 IC50 = 600 nM T49898 CC8QL6 6538940 IC50 = 1200 nM T49898 CZ5T2D 6538949 IC50 = 180 nM T49898 CSP65W 6538950 IC50 = 2800 nM T49898 C0H2JT 6538951 IC50 = 1300 nM T49898 CCG6Q1 6538952 IC50 = 3000 nM T49898 C9P5AK 6538953 IC50 = 3000 nM T49898 C1GK8C 6538954 IC50 = 4500 nM T49898 C4K9FC 6538955 IC50 = 2500 nM T49898 CUFR51 6538960 IC50 = 430 nM T49898 C5KW8Q 6538961 IC50 = 60 nM T49898 C6IWQ1 6538962 IC50 = 200 nM T49898 C0RCH9 6538963 IC50 = 300 nM T49898 CX2TI8 6538964 IC50 = 150 nM T49898 CXV4N7 6538965 IC50 = 400 nM T49898 CYCI38 6538966 IC50 = 200 nM T49898 C13IWP 6538967 IC50 = 200 nM T49898 CAO4T9 6538968 IC50 = 200 nM T49898 C1NY5R 6538969 IC50 = 60 nM T49898 CT9XA5 6539010 IC50 = 5 nM T49898 C0L5BW 6539026 IC50 = 6 nM T49898 CW9MN4 6539027 IC50 = 15 nM T49898 C60GSI 6539616 IC50 = 126 nM T49898 C3LX4A 6539618 IC50 = 501 nM T49898 CK4D8T 6539619 IC50 = 398 nM T49898 CN91SM 6539620 IC50 = 398 nM T49898 C7DR8V 6539621 IC50 = 501 nM T49898 CA5EJ9 6539622 IC50 = 794 nM T49898 C0FZA1 6539623 IC50 = 501 nM T49898 C2XC5V 6603989 IC50 = 800 nM T49898 CJ4U3H 6610355 IC50 = 2000 nM T49898 CG17TN 6914611 IC50 = 100 nM T49898 C7E2QK 6914613 IC50 > 10000 nM T49898 CL47HK 9795307 IC50 > 1000000 nM T49898 C59THZ 9802862 IC50 = 2800000 nM T49898 CH6E5L 9821686 IC50 = 20000 nM T49898 C1E2DV 9826083 IC50 > 10000 nM T49898 C6SN4V 9840475 IC50 = 400000 nM T49898 CZ9MB2 9843864 Ki = 246 nM T49898 CKL02D 9847304 IC50 = 1610 nM T49898 CE15KX 9847909 IC50 = 10 nM T49898 C16VXB 9863538 IC50 = 21 nM T49898 CRC65X 9863786 IC50 > 25000 nM T49898 CA5GN3 9864131 IC50 = 70000 nM T49898 CVC19B 9864175 IC50 = 65000 nM T49898 C7J9MI 9865229 IC50 = 270000 nM T49898 COH9E4 9885440 IC50 = 290000 nM T49898 C6L4EP 9889902 IC50 = 0.1 nM T49898 C61VZB 9906048 IC50 = 400000 nM T49898 C5BSO0 9908026 IC50 = 687 nM T49898 C7JGW4 9910100 IC50 = 33 nM T49898 CNVC67 9910699 IC50 > 100000 nM T49898 CFA49P 9910872 IC50 = 808 nM T49898 C5B2PS 9928007 IC50 = 9000000 nM T49898 C3GU2L 9928932 IC50 = 430000000 nM T49898 CQD2W7 9935079 IC50 = 1251 nM T49898 C0U6EJ 9949448 IC50 = 80 nM T49898 C2Y3FJ 9950140 IC50 = 4300000 nM T49898 C57URF 9951265 IC50 = 80 nM T49898 C2VZ4R 9951641 IC50 = 28 nM T49898 CD5M3J 9952008 IC50 = 20 nM T49898 CSRU93 9975630 IC50 = 971 nM T49898 CTU1O9 9979700 Ki = 14 nM T49898 CDHT89 9999155 Ki = 181 nM T49898 CCJ93T 9999811 IC50 = 344 nM T49898 C26QHZ 10005638 IC50 > 10000 nM T49898 C2FX0W 10023660 IC50 = 210 nM T49898 CCQ5A6 10023782 Ki = 1530 nM T49898 CVE1W8 10024433 Ki = 1894 nM T49898 CBF3T6 10043847 IC50 = 60 nM T49898 CYT3Z6 10045499 Ki = 1108 nM T49898 CV2Y8H 10051869 IC50 < 250 nM T49898 C18DAI 10069391 Ki = 278 nM T49898 C8M6PN 10092661 IC50 = 6000 nM T49898 CZP6U0 10110571 IC50 = 40 nM T49898 C50QLR 10110675 IC50 = 28 nM T49898 CK0WI8 10111486 IC50 = 230000 nM T49898 CXBW34 10114553 IC50 = 42 nM T49898 CGT4F0 10134861 IC50 = 50 nM T49898 CL2F5J 10135889 IC50 = 12 nM T49898 CPT91S 10138993 IC50 = 150 nM T49898 CZJI60 10141037 IC50 > 10000 nM T49898 C94WRY 10143231 IC50 > 10000 nM T49898 CREM37 10151881 IC50 = 1900 nM T49898 C08VYL 10158127 IC50 = 34 nM T49898 C68GUB 10159114 IC50 = 67 nM T49898 C6ZN1W 10162454 IC50 = 5000000 nM T49898 CLE8V6 10182312 IC50 = 47 nM T49898 C5Y9PK 10183407 IC50 = 19 nM T49898 CW2Y7N 10200092 IC50 = 60 nM T49898 CIGT47 10202305 IC50 = 40 nM T49898 CVRO56 10204194 IC50 = 22 nM T49898 C5P8JC 10206423 IC50 = 4428 nM T49898 CGOT91 10207821 IC50 = 240 nM T49898 C0R5AX 10215912 IC50 = 454 nM T49898 CI8MW4 10216627 IC50 = 870 nM T49898 CEW30I 10217590 IC50 > 50000 nM T49898 CHM97B 10221628 IC50 = 50 nM T49898 C84VWO 10221806 IC50 = 450 nM T49898 CLW0H7 10223662 IC50 = 40 nM T49898 C1KX3P 10248401 Ki > 10000 nM T49898 CE19JD 10249602 Ki = 1638 nM T49898 CJ1AN4 10251513 Ki = 43 nM T49898 CNQH37 10253652 IC50 = 2500 nM T49898 CZ6EK3 10269548 IC50 = 240000 nM T49898 CG65JV 10275574 IC50 = 200 nM T49898 CG56FT 10277583 IC50 = 232 nM T49898 C58NEO 10295144 IC50 = 160 nM T49898 C85MHR 10297090 IC50 = 60 nM T49898 C6PL7N 10297469 IC50 = 60 nM T49898 C6J7FS 10297929 IC50 = 63 nM T49898 CRAB41 10317147 IC50 = 1108 nM T49898 CKNL70 10319097 Ki = 28 nM T49898 C9J3RM 10320107 Ki = 851 nM T49898 C6USY4 10339994 IC50 = 100 nM T49898 CMY9D2 10340715 Ki > 10000 nM T49898 CTX01B 10341351 IC50 = 1240 nM T49898 C6MIL0 10362606 IC50 = 10 nM T49898 CVN8T9 10379252 IC50 = 160 nM T49898 C0UJ5R 10389002 IC50 > 10000 nM T49898 CA8B5T 10390073 IC50 > 10000 nM T49898 CP5IH6 10390085 IC50 > 10000 nM T49898 CH8KM7 10414039 IC50 = 250 nM T49898 C2B0IU 10421236 IC50 = 2500 nM T49898 C10NPZ 10429133 IC50 = 8000 nM T49898 CC3L8Z 10430000 Ki = 3925 nM T49898 C2Z6NO 10431144 IC50 = 330 nM T49898 CFLH53 10432113 IC50 > 10000 nM T49898 CFNM76 10434333 Ki = 1667 nM T49898 CHB2D8 10449125 Ki = 5841 nM T49898 CL7PF2 10451087 IC50 > 10000 nM T49898 CH4CY9 10471016 IC50 = 30000 nM T49898 CXCO41 10479319 Ki = 5 nM T49898 CKV93A 10493297 IC50 = 25000 nM T49898 C8QN3B 10504063 IC50 = 1300 nM T49898 CFIY95 10504197 IC50 = 5300 nM T49898 CZAF27 10512545 IC50 = 50000 nM T49898 C1DVX0 10520326 IC50 = 8000 nM T49898 C21BTO 10524103 IC50 > 100000 nM T49898 CKA05R 10554185 IC50 = 10000 nM T49898 C0ZTJ9 10572551 IC50 > 1000000 nM T49898 CEKB07 10596901 IC50 = 1800 nM T49898 CTM8Q3 10597689 IC50 = 350 nM T49898 CJ69GO 10598282 IC50 > 1000000 nM T49898 CWYE93 10615524 IC50 = 2400 nM T49898 CKX2L8 10623869 IC50 = 10000 nM T49898 CW2K9B 10634429 IC50 = 10000 nM T49898 C4T3MI 10634685 IC50 = 40000 nM T49898 CQV3H7 10645840 IC50 = 430 nM T49898 CG1S7F 10645935 IC50 = 2300 nM T49898 CP76GB 10647476 IC50 = 10000 nM T49898 C48AXV 10647526 IC50 = 1300 nM T49898 C0BI5S 10658427 IC50 = 40000 nM T49898 C8A3EI 10671123 IC50 > 1000000 nM T49898 CW2XK8 10671675 IC50 = 4300 nM T49898 C3LHP0 10693555 IC50 = 850 nM T49898 C5ZHX0 10694163 IC50 = 430 nM T49898 CNB06C 10694961 IC50 = 4200 nM T49898 C2MRA7 10716972 IC50 > 1000000 nM T49898 C2YM5I 10717330 IC50 = 300 nM T49898 C0W8ED 10733091 IC50 = 17000 nM T49898 CZ2B5D 10738939 IC50 = 620000 nM T49898 CE2FZ5 10763151 IC50 > 1000000 nM T49898 C38HVX 10764739 IC50 = 7200 nM T49898 CX70VJ 10765267 IC50 = 4000 nM T49898 CL9H2N 10786933 IC50 = 300 nM T49898 C3F4DW 10802411 IC50 = 65000 nM T49898 C7MJ0P 10807095 IC50 = 1100 nM T49898 CHJP65 10815297 IC50 = 1000 nM T49898 C39CYP 10836574 IC50 = 800 nM T49898 CU9V1B 10837228 IC50 > 1000000 nM T49898 CBOP58 11293798 Ki > 10000 nM T49898 C29IST 11302358 IC50 = 3700 nM T49898 C26BZX 11362471 Ki > 10000 nM T49898 CWXB93 11397177 Ki > 10000 nM T49898 CWM18I 11406175 IC50 > 50000 nM T49898 C1WXC5 11417488 IC50 > 50000 nM T49898 C1F9NV 11419598 IC50 = 3600 nM T49898 CU0MY9 11464906 IC50 = 4100 nM T49898 CXT91K 11488074 IC50 = 4300 nM T49898 CL1WN3 11518075 IC50 = 50 nM T49898 C1RCA9 11525251 IC50 = 1070 nM T49898 C0X2AS 11533897 IC50 = 1550 nM T49898 CTG83F 11539329 Ki > 8900 nM T49898 C1W5OC 11562531 IC50 = 1660 nM T49898 C72XAP 11569937 IC50 = 466 nM T49898 CD3E8M 11574606 IC50 = 140 nM T49898 CMIL86 11590363 Ki > 8900 nM T49898 C2V0DP 11598432 IC50 = 494 nM T49898 C5B3XJ 11620410 IC50 > 40000 nM T49898 CIWA03 11632150 Ki = 706 nM T49898 C9T6SC 11640926 Ki > 8900 nM T49898 CEV5X2 11646645 Ki = 240 nM T49898 C2CVI7 11647020 Ki = 1224 nM T49898 CQKD95 11669987 IC50 = 12 nM T49898 CYM9A8 11678367 IC50 = 1340 nM T49898 C93KHF 11718021 Ki = 367 nM T49898 CLZU92 11739898 IC50 = 1500 nM T49898 CR93CE 11743030 Ki = 17 nM T49898 CJSV21 11744184 Ki > 10000 nM T49898 CYZ87D 11774496 IC50 = 14 nM T49898 CE6X7A 11792319 IC50 = 300 nM T49898 C4V7JE 11794083 IC50 = 1000 nM T49898 C6N0RY 11974955 Ki > 10000 nM T49898 CNIK34 11974956 Ki > 10000 nM T49898 C0YX7V 11974957 Ki > 10000 nM T49898 CLTK95 11975073 Ki = 193 nM T49898 CDP24B 11975074 Ki = 133 nM T49898 CXR6J8 11975075 Ki = 38 nM T49898 C2QV6O 11975201 Ki > 10000 nM T49898 CAP2M7 11975202 Ki > 10000 nM T49898 C5XWU4 11975203 Ki = 1259 nM T49898 CZF8T4 11975204 Ki = 6615 nM T49898 CX2AS7 11975205 Ki = 2500 nM T49898 C3OHQ1 11975206 Ki = 14 nM T49898 C8E4TS 11992146 IC50 = 30000 nM T49898 CND6F5 12084804 IC50 = 500000 nM T49898 C7RLP2 12084805 IC50 = 420000 nM T49898 CNJ7P6 12084806 IC50 = 10000000 nM T49898 C52MGL 12084807 IC50 = 2700000 nM T49898 CV05BZ 12084808 IC50 = 600000 nM T49898 CMJ1S2 12084809 IC50 = 130000 nM T49898 CG1F0S 12084810 IC50 = 100000 nM T49898 C5E0CK 12084811 IC50 = 500000 nM T49898 CVAW53 12084812 IC50 = 52000000 nM T49898 CPTF05 12084813 IC50 = 100000 nM T49898 CJR7W4 13521419 IC50 = 10000 nM T49898 CES1T9 13908780 IC50 > 1000000 nM T49898 C2Z8DQ 14624081 IC50 = 100 nM T49898 C7N6CQ 15604547 IC50 = 22 nM T49898 C15QHL 15693435 IC50 = 12000 nM T49898 CP8OW6 15858662 IC50 = 43000 nM T49898 CP5AC1 15942652 IC50 = 130 nM T49898 C3CPB2 16007031 IC50 = 10000 nM T49898 CFPW41 16007116 Ki > 8900 nM T49898 C1DO0X 16037278 IC50 = 19800 nM T49898 C7BS2R 16037674 IC50 > 10000 nM T49898 CB2H4D 16037675 IC50 = 600 nM T49898 C9TU1O 16046126 IC50 = 1 nM T49898 C15QAG 16113377 IC50 = 11 nM T49898 C5GZ4J 16113378 IC50 = 5 nM T49898 C1O9SF 16113484 IC50 = 2 nM T49898 CU01IX 16409607 IC50 = 90000 nM T49898 CAK1C4 16666757 IC50 > 100000 nM T49898 C1QRG8 16666806 IC50 > 100000 nM T49898 CJ9C7N 16666859 IC50 > 100000 nM T49898 C5JQ6H 16666860 IC50 > 100000 nM T49898 C4VW0O 16666861 IC50 > 100000 nM T49898 C1IO4K 16666862 IC50 > 100000 nM T49898 CS1LR2 16666908 IC50 > 100000 nM T49898 CI32LX 16666909 IC50 = 13300 nM T49898 C07BIL 16666910 IC50 > 100000 nM T49898 C71TSX 16666911 IC50 > 100000 nM T49898 CUR7H3 16719862 IC50 = 18000 nM T49898 CP1RF4 16739311 IC50 = 1540 nM T49898 C3YNI9 16746003 IC50 = 230000 nM T49898 CPH09W 16746013 IC50 = 5000000 nM T49898 C08CHX 16746085 IC50 = 30000 nM T49898 CD27OV 16746115 IC50 = 530000 nM T49898 CF8RA0 16746116 IC50 = 300000 nM T49898 CES7Z0 16746117 IC50 = 900000 nM T49898 C90JGS 17312697 IC50 = 1400 nM T49898 CZ90RF 18516895 IC50 = 470 nM T49898 CHVU30 18516919 IC50 = 2000 nM T49898 CQO3F4 18516938 IC50 = 4800 nM T49898 CFAY17 18516981 IC50 = 5700 nM T49898 C59CVU 19689599 IC50 = 35 nM T49898 CZ06SD 20668980 IC50 = 2800000 nM T49898 CENP10 21039972 IC50 = 32 nM T49898 CKV09C 21817592 IC50 = 2100 nM T49898 C3DJ7X 21868318 IC50 > 500000 nM T49898 C13WHU 21980365 IC50 = 250 nM T49898 C39NXD 21980383 IC50 = 30 nM T49898 C75ZLY 21980427 IC50 = 250 nM T49898 CD7YS1 21980580 IC50 < 250 nM T49898 CQI80X 21980631 IC50 = 250 nM T49898 CP7BE6 21980647 IC50 = 200 nM T49898 C13NVO 21980695 IC50 = 250 nM T49898 CE93IF 21980705 IC50 = 250 nM T49898 CA24TJ 21980718 IC50 = 250 nM T49898 CM37OL 21980722 IC50 = 30 nM T49898 CQ4G1U 21988176 IC50 = 40 nM T49898 CIV7G5 21988177 IC50 = 450 nM T49898 CJ4G1H 21988178 IC50 = 39 nM T49898 CH27DF 21988185 IC50 = 560 nM T49898 C0DW3O 21988189 IC50 = 600 nM T49898 C18WFG 21988212 IC50 = 31 nM T49898 COH4Y2 21988214 IC50 = 700 nM T49898 C6QU7C 21988217 IC50 = 85 nM T49898 CGJ6I9 21988220 IC50 = 160 nM T49898 CQ3P5M 21988222 IC50 = 140 nM T49898 CIX64M 21988223 IC50 = 28 nM T49898 C6A8DH 21988224 IC50 = 330 nM T49898 C8CGO6 21988247 IC50 = 440 nM T49898 CXI0N7 21988261 IC50 = 90 nM T49898 CUK89W 21988265 IC50 = 450 nM T49898 C0IR2S 21988310 IC50 = 550 nM T49898 CWDZ32 21988320 IC50 = 380 nM T49898 C69CDM 21988326 IC50 = 150 nM T49898 CB5SV4 21988329 IC50 = 30 nM T49898 CL87NE 22061088 IC50 > 1000 nM T49898 CNYQ64 23074669 IC50 = 260000 nM T49898 CPL7J5 23635674 IC50 = 29 nM T49898 C6YF5D 23645577 IC50 = 3400 nM T49898 C95CXB 23645579 IC50 = 5600 nM T49898 CHK57M 23645580 IC50 = 16000 nM T49898 CQHK69 23646624 IC50 = 1600 nM T49898 C2JTA3 23647573 IC50 = 4900 nM T49898 C17HUI 23647581 IC50 = 3400 nM T49898 C3JWK1 23654166 IC50 = 250 nM T49898 CA3I4T 24753787 IC50 > 50000 nM T49898 C60JXM 24780352 IC50 < 1 nM T49898 CCP2M3 24822704 IC50 > 50000 nM T49898 CZ48LS 24825971 IC50 > 50000 nM T49898 CP5EL9 24884696 IC50 = 250 nM T49898 CTFS94 24884697 IC50 < 250 nM T49898 C70ZFW 24884912 IC50 > 10000 nM T49898 C4V9GI 24960018 IC50 > 50000 nM T49898 CD18LU 24970432 IC50 = 13000 nM T49898 CTKL39 24970435 IC50 = 9000 nM T49898 C9M1IV 24970438 IC50 = 150 nM T49898 CX1HL8 25032704 Ki > 8910 nM T49898 CHLQ49 25063262 IC50 > 100000 nM T49898 C2CXU0 25164676 Ki = 5.012 nM T49898 CP28KV 25176840 IC50 = 130 nM T49898 C6FGQ1 25206346 IC50 = 3700 nM T49898 CLB28U 25271180 IC50 > 100000 nM T49898 CGHR32 25271181 IC50 > 100000 nM T49898 C3E9XU 25271513 IC50 > 100000 nM T49898 CGBX14 25271514 IC50 > 100000 nM T49898 C76NWM 25271515 IC50 > 100000 nM T49898 C6C4YR 25271516 IC50 > 100000 nM T49898 CUAK50 25271517 IC50 > 100000 nM T49898 CIR67H 25271518 IC50 > 100000 nM T49898 CC71QJ 27666048 IC50 > 100000 nM T49898 CUF71P 42066883 IC50 = 2900 nM T49898 CPBZ35 42610232 IC50 > 100000 nM T49898 CU9E4P 42629114 IC50 = 4600 nM T49898 CLW80F 44160269 IC50 = 26000 nM T49898 CJ7AF4 44203948 IC50 = 7500 nM T49898 CG8CQ2 44315777 IC50 = 40000 nM T49898 C9E8ZL 44315861 IC50 = 6000000 nM T49898 CX07HO 44315870 IC50 = 7000000 nM T49898 CCW6U1 44315871 IC50 = 5300000 nM T49898 CTBN92 44315885 IC50 = 6500000 nM T49898 C6GS3M 44315921 IC50 = 220000 nM T49898 CNRD64 44315922 IC50 = 33000000 nM T49898 C7Y2TH 44315925 IC50 = 230000 nM T49898 CEJ2I1 44315926 IC50 = 170000 nM T49898 C6DP8U 44315927 IC50 = 160000 nM T49898 CQ23YJ 44315928 IC50 = 130000 nM T49898 C7PRE3 44315929 IC50 = 45000 nM T49898 CF45UQ 44315940 IC50 = 210000 nM T49898 C2Z1BS 44315980 IC50 = 400000 nM T49898 C0VZ8W 44315981 IC50 = 360000 nM T49898 C8MS5V 44315985 IC50 = 300000 nM T49898 CFT6X9 44315986 IC50 = 800000 nM T49898 C13ITU 44316008 IC50 = 4000000 nM T49898 CRI1G0 44316009 IC50 = 3000000 nM T49898 C3H8RI 44316010 IC50 = 10800000 nM T49898 CV5C8N 44316102 IC50 = 4400000 nM T49898 C27WIA 44316103 IC50 = 1300000 nM T49898 CFDS19 44316108 IC50 = 9000000 nM T49898 C5MW0R 44316109 IC50 = 7000000 nM T49898 CB0UX1 44316124 IC50 = 5000000 nM T49898 C4NO8K 44316125 IC50 = 5000000 nM T49898 CH8T1V 44316130 IC50 = 5000000 nM T49898 CE50IV 44316136 IC50 = 1400000 nM T49898 CIR0V5 44316137 IC50 = 1300000 nM T49898 C5LPT1 44316145 IC50 = 5000000 nM T49898 CPF5S0 44316151 IC50 = 1000000 nM T49898 CMI19E 44316152 IC50 = 790000 nM T49898 CRB3X0 44316153 IC50 = 80000 nM T49898 C07QCT 44316154 IC50 = 1300000 nM T49898 CL0YW6 44316169 IC50 = 1200000 nM T49898 C2BJ9Q 44316171 IC50 = 1200000 nM T49898 C2NIF5 44316180 IC50 = 1200000 nM T49898 C3R4GW 44316183 IC50 = 250000 nM T49898 CLP32H 44316192 IC50 = 10000000 nM T49898 CAW13E 44316198 IC50 = 500000 nM T49898 C8B3FK 44316199 IC50 = 500000 nM T49898 CPB41O 44316289 IC50 = 2300000 nM T49898 C3JYD0 44316290 IC50 = 1600000 nM T49898 C7WC3U 44316293 IC50 = 450000 nM T49898 CIFR71 44316294 IC50 = 5000000 nM T49898 CQI1M5 44316332 IC50 = 1500000 nM T49898 C8T3FO 44316339 IC50 = 10000000 nM T49898 C4LZM2 44316489 IC50 = 700000 nM T49898 C0FY9X 44316518 IC50 = 560000 nM T49898 CWH8Z1 44321838 IC50 > 1000000 nM T49898 CMD5V4 44321840 IC50 > 1000000 nM T49898 CSB0Y5 44322128 IC50 > 1000000 nM T49898 CF7T3B 44322130 IC50 > 1000000 nM T49898 C2PI0F 44322155 IC50 > 1000000 nM T49898 CBA6K4 44332160 IC50 = 16000 nM T49898 CJEP87 44332387 IC50 > 100000 nM T49898 CHK0B9 44332407 IC50 = 14000 nM T49898 C93HEX 44332604 IC50 = 10000 nM T49898 C81VKL 44332664 IC50 = 30 nM T49898 CY2X1B 44332666 IC50 = 13000 nM T49898 CL2TC5 44332685 IC50 > 100000 nM T49898 C1KSW5 44335197 IC50 > 10000 nM T49898 C0KD4U 44346053 IC50 > 10000 nM T49898 CG9P2I 44353519 IC50 = 1000 nM T49898 C46QZL 44353529 IC50 = 330 nM T49898 CO5TD3 44353560 IC50 = 400 nM T49898 C5PIG4 44353568 IC50 = 300 nM T49898 C2P4VE 44353607 IC50 = 500 nM T49898 CF1A2K 44353670 IC50 = 6000 nM T49898 C84YDA 44353701 IC50 = 300000 nM T49898 C1LYR2 44353706 IC50 = 900 nM T49898 C2ZL8B 44353713 IC50 > 1000000 nM T49898 CHP67O 44353737 IC50 > 1000000 nM T49898 C45EFJ 44353766 IC50 = 130000 nM T49898 CAYU92 44353854 IC50 = 300 nM T49898 CYV2D7 44368815 IC50 > 10000 nM T49898 C75NGL 44384514 IC50 > 10000 nM T49898 CV0F4D 44384547 IC50 = 47000 nM T49898 CQF8Y7 44384548 IC50 > 10000 nM T49898 CF01AV 44384717 IC50 = 120 nM T49898 CE0J2Q 44384882 IC50 = 250 nM T49898 C1HQR9 44384929 IC50 = 310 nM T49898 CI2L9R 44384964 IC50 > 10000 nM T49898 CC09FT 44384965 IC50 = 82500 nM T49898 CE9PU7 44385035 IC50 > 10000 nM T49898 C15SOY 44385064 IC50 = 41 nM T49898 CQGW07 44385080 IC50 > 100000 nM T49898 CH4GJ3 44385083 IC50 = 550 nM T49898 CL4Y9M 44385116 IC50 = 33000 nM T49898 C8YNC3 44385264 IC50 = 80 nM T49898 C64LMY 44385265 IC50 = 39 nM T49898 CY87KD 44385687 IC50 = 1000 nM T49898 C82JNP 44385691 IC50 = 350 nM T49898 CUI34C 44385739 IC50 = 90000 nM T49898 C9XW3C 44385797 IC50 = 230 nM T49898 C61PAS 44385804 IC50 = 150 nM T49898 C8EIN0 44387663 IC50 > 10000 nM T49898 CSOU41 44401258 IC50 > 1000 nM T49898 CD4Y6K 44401272 IC50 = 126 nM T49898 CXVJ24 44401282 IC50 = 392 nM T49898 C4MCG6 44401283 IC50 = 77 nM T49898 CL7F2K 44401284 IC50 = 4 nM T49898 CN7H9W 44401286 IC50 = 43 nM T49898 CDC73G 44401340 IC50 = 22 nM T49898 CJHM62 44401365 IC50 = 135 nM T49898 CG4X5Z 44401370 IC50 = 15 nM T49898 CY2HX9 44401389 IC50 = 160 nM T49898 CB5M3L 44401397 IC50 = 9 nM T49898 CUY8A3 44401410 IC50 = 10 nM T49898 C6OR3S 44401412 IC50 = 9 nM T49898 C0IH5E 44401413 IC50 = 252 nM T49898 CS9V3J 44401429 IC50 = 34 nM T49898 C8L5ZH 44401437 IC50 = 0.9 nM T49898 CBY03Q 44401438 IC50 = 34 nM T49898 C7BWI1 44401485 IC50 > 1000 nM T49898 CV0X6H 44401486 IC50 = 4 nM T49898 CIB5V1 44401506 IC50 = 11 nM T49898 CN9WJ5 44401507 IC50 = 4 nM T49898 C1JGB5 44401511 IC50 = 15 nM T49898 C9WZ5P 44401512 IC50 > 1000 nM T49898 CQHB30 44401517 IC50 = 25 nM T49898 C6A2LQ 44401518 IC50 = 2 nM T49898 C3P0SZ 44401555 IC50 > 1000 nM T49898 C5C3BG 44401556 IC50 = 8 nM T49898 C7JD9F 44401574 IC50 > 1000 nM T49898 CXW7Y1 44401575 IC50 = 10 nM T49898 C48GXY 44401597 IC50 = 32 nM T49898 CWX5P3 44401602 IC50 = 248 nM T49898 C2EBH4 44401603 IC50 > 1000 nM T49898 CW56HM 44401628 IC50 > 1000 nM T49898 CQK0M1 44401667 IC50 > 1000 nM T49898 CO8C7T 44401668 IC50 = 562 nM T49898 CV7N5S 44401669 IC50 = 430 nM T49898 C9V5GQ 44401670 IC50 = 3 nM T49898 CAN72B 44408691 IC50 = 8800 nM T49898 CWM75V 44412739 IC50 = 1410 nM T49898 C5HZF2 44413509 IC50 = 24 nM T49898 C3D4FG 44413527 IC50 > 1000 nM T49898 CETQ79 44427518 IC50 > 50000 nM T49898 COPG94 44427519 IC50 > 10000 nM T49898 C2U5KW 44430873 IC50 = 6200 nM T49898 C0P8BA 44430874 IC50 = 9000 nM T49898 CQXL12 44430875 IC50 = 6500 nM T49898 C25WQT 44430876 IC50 = 2100 nM T49898 C9I2GJ 44430877 IC50 = 2000 nM T49898 CKCX40 44430878 IC50 = 4200 nM T49898 C0ZXY6 44430879 IC50 = 3300 nM T49898 CL7C6R 44430880 IC50 = 3300 nM T49898 CS9O6C 44430882 IC50 > 10000 nM T49898 C98QBK 44430883 IC50 > 10000 nM T49898 CD8B4J 44430884 IC50 > 10000 nM T49898 C7PNC9 44430885 IC50 > 10000 nM T49898 CY6P9J 44430886 IC50 > 10000 nM T49898 C8MLH2 44430887 IC50 > 10000 nM T49898 CNU34S 44430906 IC50 = 1600 nM T49898 CLEX18 44430913 IC50 = 410 nM T49898 CZIC28 44430916 IC50 = 1500 nM T49898 C2J5XB 44430917 IC50 = 2000 nM T49898 CBQM21 44430920 IC50 = 1900 nM T49898 CQ7L8Y 44430921 IC50 = 560 nM T49898 CDW6L0 44430924 IC50 = 2700 nM T49898 CXK2J8 44430925 IC50 = 1700 nM T49898 CA0N4B 44430927 IC50 = 1100 nM T49898 CQN31M 44430929 IC50 = 5600 nM T49898 CL7X4E 44430931 IC50 = 21000 nM T49898 CG4E1T 44431447 IC50 = 1040 nM T49898 C5QWY4 44431448 IC50 = 1060 nM T49898 CP76WK 44431449 IC50 = 1140 nM T49898 CR1G5K 44431450 IC50 = 461 nM T49898 CJ64DM 44431451 IC50 = 439 nM T49898 C0XFS5 44431452 IC50 = 48 nM T49898 C5VPN4 44431453 IC50 = 540 nM T49898 CE81LF 44431454 IC50 = 847 nM T49898 CGK6T3 44431455 IC50 = 1770 nM T49898 C0NZX8 44431456 IC50 = 334 nM T49898 CE7N4S 44431457 IC50 = 781 nM T49898 C4R6AN 44431460 IC50 = 180 nM T49898 CJM89C 44431461 IC50 = 1240 nM T49898 CB9RV2 44447912 IC50 = 30 nM T49898 C4MQJ7 44447913 IC50 = 80 nM T49898 C2N6CE 44447930 IC50 = 28 nM T49898 C48HGY 44517741 IC50 = 0.8 nM T49898 CA7TD4 44517742 IC50 = 1 nM T49898 C4WRN5 44541014 IC50 = 39.2 nM T49898 C3VRO9 44557921 IC50 > 10000 nM T49898 C1A4XG 44562420 IC50 > 100000 nM T49898 C3UV2W 44562431 IC50 > 100000 nM T49898 CWN43A 44562683 IC50 = 11 nM T49898 CE7LN0 44562736 IC50 = 120 nM T49898 C6PJI0 44562737 IC50 = 100 nM T49898 C8C6AW 44562738 IC50 = 9 nM T49898 C1VQ2B 44563116 IC50 = 71 nM T49898 CP5GJ1 44563117 IC50 = 180 nM T49898 CS19XE 44563151 IC50 = 150 nM T49898 CM0GJ1 44563897 IC50 = 50000 nM T49898 CTB96Y 44579918 IC50 > 100000 nM T49898 C28QLM 44605035 IC50 > 50000 nM T49898 C75XHS 44605037 IC50 > 50000 nM T49898 C8ZCP1 44631900 IC50 = 11 nM T49898 C2I3QV 45267582 IC50 = 25 nM T49898 C7H0EZ 45267583 IC50 = 6330 nM T49898 C9V6NQ 45267633 IC50 = 26 nM T49898 CNA6Z4 45267641 IC50 = 3090 nM T49898 C75WAC 45268471 IC50 = 2730 nM T49898 CL3ZD2 45268500 IC50 = 25 nM T49898 C43MRK 45268501 IC50 = 2600 nM T49898 C8WJ4I 45268513 IC50 = 52 nM T49898 CN4TD8 45269319 IC50 = 250 nM T49898 C0L3KN 45269326 IC50 = 2040 nM T49898 CH59DU 45269365 IC50 = 3170 nM T49898 CVJ70Z 45269366 IC50 = 64 nM T49898 C9NCR0 45269376 IC50 = 81 nM T49898 C6B9VH 45270159 IC50 = 10800 nM T49898 C59YDL 45271022 IC50 = 3100 nM T49898 CG83KW 45271845 IC50 = 200 nM T49898 C92ZKY 45271846 IC50 = 390 nM T49898 C4C0TD 45271854 IC50 = 10900 nM T49898 C6U1LK 45271859 IC50 = 7920 nM T49898 C04AVC 45271879 IC50 = 360 nM T49898 C0KFU4 45271889 IC50 = 2700 nM T49898 CK3F4V 45272705 IC50 = 5 nM T49898 CT7RV8 45272713 IC50 = 2210 nM T49898 C06JQE 45273683 IC50 = 146 nM T49898 C6E2SC 45482700 IC50 > 10000 nM T49898 CZXH74 45482750 IC50 > 10000 nM T49898 CY3HW5 46224684 IC50 = 320 nM T49898 C1J6GR 46224908 IC50 > 10000 nM T49898 CYT37A 46232443 IC50 > 50000 nM T49898 C48ZVW 46232555 IC50 > 50000 nM T49898 CS9B1U 46232556 IC50 > 50000 nM T49898 CC2WT4 46232590 IC50 = 200 nM T49898 CGO1J5 46830766 Ki = 909 nM T49898 CF7HK2 46830767 Ki = 769 nM T49898 C2HJ1X 46830768 Ki > 10000 nM T49898 CLS29B 46872626 IC50 > 10000 nM T49898 CJOM49 46880136 IC50 = 28400 nM T49898 CQ7ET6 46881853 IC50 = 2500 nM T49898 C29PHE 46882055 IC50 = 220 nM T49898 C2O8RZ 46886323 IC50 > 1000 nM T49898 CP34VL 46929748 IC50 > 1000 nM T49898 CKL1V8 49798556 IC50 > 20000 nM T49898 CKYX24 49830272 Ki = 39.81 nM T49898 CVM6X8 49830280 Ki > 10000 nM T49898 C3X6DN 49830474 Ki > 10000 nM T49898 CCL3R5 49867929 IC50 = 14000 nM T49898 CEQN27 52936621 Ki > 1000 nM T49898 C8BOP9 52942870 IC50 = 15 nM T49898 C0K5NI 52944208 IC50 = 2900 nM T49898 CO1TP3 52947886 IC50 = 55 nM T49898 CH2O0D 52948241 IC50 = 5000 nM T49898 CY8V0Q 52949108 IC50 = 104 nM T49898 CBR69H 53695812 IC50 = 10000 nM T49898 CVI9A5 53788948 IC50 = 20 nM T49898 CJ9GH5 54339282 IC50 = 330 nM T49898 CK85QR 54373950 IC50 = 10000 nM T49898 C2G3AY 54726684 IC50 > 100000 nM T49898 CR50TJ 56835147 IC50 = 10000 nM T49898 CPHX64 57325478 IC50 > 50000 nM T49898 CQ9BW4 57325479 IC50 > 50000 nM T49898 C5YRF8 57328039 IC50 = 22 nM T49898 CP7UB8 57383477 IC50 = 500 nM T49898 CS72WD 58015961 IC50 > 1600 nM T49898 CVK0G4 58056356 IC50 > 50000 nM T49898 C1MR8Q 60097495 IC50 > 10000 nM T49898 CK0XR7 66560844 IC50 = 2000 nM T49898 CR2T5Q 66934034 Ki < 100 nM T49898 C59ZIA 67284569 IC50 = 75 nM T49898 CYI75G 68678653 IC50 > 30000 nM T49898 C3NVZ6 70681070 IC50 = 1200 nM T49898 C56ZER 70681071 IC50 = 150 nM T49898 CV24XU 70681532 IC50 = 240 nM T49898 CRYW49 70681533 IC50 = 700 nM T49898 C1R6HY 70683192 IC50 = 24 nM T49898 C3NCF2 70683641 IC50 = 180 nM T49898 CY51SV 70683642 IC50 = 200 nM T49898 C6QZ5U 70685271 IC50 = 10 nM T49898 CPTG79 70685272 IC50 = 390 nM T49898 C4PW8O 70685778 IC50 = 1100 nM T49898 CN3E5T 70685779 IC50 = 1700 nM T49898 C6DAJ0 70687420 IC50 = 16 nM T49898 C6FO8B 70687421 IC50 = 47 nM T49898 C01WIM 70689476 IC50 = 21 nM T49898 CAE31H 70689940 IC50 = 28 nM T49898 C1IN7G 70689941 IC50 = 330 nM T49898 CS1G5L 70691585 IC50 = 24 nM T49898 CDWB98 70691595 IC50 = 19 nM T49898 C5MT8A 70691596 IC50 = 1700 nM T49898 CC5A4K 70692098 IC50 = 6 nM T49898 CADI76 70692099 IC50 = 1300 nM T49898 CW9MY1 70693675 IC50 = 50 nM T49898 C2L6OP 70693678 IC50 = 13 nM T49898 CNRC67 70693679 IC50 = 40 nM T49898 CJZ5E1 70693680 IC50 = 150 nM T49898 C2QJ8X 70695789 IC50 = 38 nM T49898 CPW57H 70695790 IC50 = 15 nM T49898 CC8WG5 70695791 IC50 = 24 nM T49898 C2UMZ0 70695792 IC50 = 41 nM T49898 C1SX4Q 70695793 IC50 = 10 nM T49898 C76JFM 70696269 IC50 = 10000 nM T49898 CNI64Y 70696270 IC50 = 1400 nM T49898 CK58RV 71449587 IC50 = 62 nM T49898 C6VF7J 71453206 IC50 = 230 nM T49898 CO0WF5 71454941 IC50 = 55 nM T49898 CF74SL 71454944 IC50 = 14000 nM T49898 CZG8I6 71456727 IC50 = 36 nM T49898 CE1IX7 71456728 IC50 = 3200 nM T49898 CV28JD 71458027 IC50 = 800 nM T49898 C14OGU 71458568 IC50 = 12 nM T49898 CVQ62G 71458571 IC50 = 7.4 nM T49898 C74VKX 71458572 IC50 = 100 nM T49898 CM1ND2 71458573 IC50 = 210 nM T49898 C3S0NP 71458574 IC50 = 1200 nM T49898 CY6WI2 71458575 IC50 = 32000 nM T49898 C15XAV 71460420 IC50 = 48 nM T49898 CKV1P2 71460421 IC50 = 320 nM T49898 CT7K3A 71460422 IC50 = 1400 nM T49898 C25FQP 71462104 IC50 = 100 nM T49898 C31ZKB 71462893 IC50 = 100 nM T49898 CG2KF6 71462956 IC50 = 10000 nM T49898 CUGP02 71494949 IC50 = 7 nM T49898 CBE67N 71731769 IC50 > 10000 nM T49898 CZY98A 71817643 IC50 = 422 nM T49898 CPWR29 71817644 IC50 = 119 nM T49898 CIJ6C1 71817645 IC50 = 183 nM T49898 CK1SR0 71817646 IC50 = 58 nM T49898 C2SK0J 71817647 IC50 = 77 nM T49898 CYH53S 71817796 IC50 = 49 nM T49898 CBNL49 71817797 IC50 = 169 nM T49898 C5XKF1 71817798 IC50 = 215 nM T49898 CK2OG4 71817799 IC50 = 555 nM T49898 C6UN8B 71817800 IC50 = 777 nM T49898 C51TYM 71817954 IC50 = 23 nM T49898 CYPU34 71817955 IC50 = 93 nM T49898 CYG95S 72707651 IC50 = 610 nM T49898 CNP0V5 72707724 IC50 = 584 nM T49898 CU4A5Q 72707728 IC50 = 571 nM T49898 CZAM98 72707790 IC50 = 569 nM T49898 CP13FK 72707853 IC50 = 522 nM T49898 C95WHV 73345983 IC50 = 184 nM T49898 CAX4V9 73345984 IC50 = 100 nM T49898 CJV80N 73347509 IC50 = 90 nM T49898 CO9W2Z 73349047 IC50 = 118 nM T49898 CYP0Q6 73350609 IC50 = 152 nM T49898 C2G6XN 73350612 IC50 > 999 nM T49898 CZ13WR 73350613 IC50 = 66 nM T49898 CUG46F 73352115 IC50 = 301 nM T49898 CI79PR 73355077 IC50 = 148 nM T49898 C4D7NR 73355078 IC50 = 202 nM T49898 C3WYF7 76331558 IC50 = 700 nM T49898 C7VA5U 78161839 IC50 = 53 nM T49898 CWR57U 78357763 IC50 = 13.9 nM T49898 CQ2SU8 78673832 IC50 > 30000 nM T49898 CE0W9R 78673833 IC50 > 30000 nM T49898 C8D3XO 86765295 IC50 > 10000 nM T49898 C0GYK1 86765296 IC50 = 5300 nM T49898 CUY63S 90645193 IC50 > 10000 nM T49898 CHP58B 118329742 IC50 = 1380 nM T49898 C6OAP9 118329761 IC50 = 1660 nM T49898 CX58DI 118716791 IC50 > 30000 nM T49898 CD9X2B 118716796 IC50 > 30000 nM T49898 C2YJ0O 118716797 IC50 > 30000 nM T49898 CL3UO9 118716798 IC50 > 30000 nM T49898 C71BAM 118716799 IC50 > 30000 nM T49898 CU4EL6 118716806 IC50 > 30000 nM T49898 CSW6L2 122667245 IC50 = 20225 nM T49898 C63VIC 122667249 IC50 = 97.2 nM T49898 CEG56K 122667252 IC50 = 133.8 nM T49898 C3J9UR 122667253 IC50 = 2429.5 nM T49898 C1SDO8 122667293 IC50 = 300.9 nM T49898 CLHF95 122667296 IC50 = 35.8 nM T49898 C5R4PU 122667312 IC50 = 800.9 nM T49898 CG8ZM5 122667313 IC50 = 1671.1 nM T49898 CAQP38 122667319 IC50 = 135.5 nM T49898 CAJH71 122667328 IC50 = 150 nM T49898 CSY3M0 122667329 IC50 = 100.5 nM T49898 CJU5O4 122667350 IC50 = 139.7 nM T49898 C09GPH 122667359 IC50 = 103.1 nM T49898 CW95MK 122667361 IC50 = 44 nM T49898 CZT1C4 122667385 IC50 = 411.9 nM T49898 CR5MA6 122667387 IC50 = 230.7 nM T49898 COF75Z 126970673 IC50 = 430 nM T49898 C1SP3H 127030849 IC50 = 777 nM T49898 C4PFZ0 127046319 IC50 = 1000 nM T49898 C0CX4P 127046320 IC50 = 1000 nM T49898 CUD8G5 127046367 IC50 = 1700 nM T49898 CA83YU 127047442 IC50 = 500 nM T49898 CNJQ71 127047443 IC50 = 1000 nM T49898 CC1VO7 127047444 IC50 > 25000 nM T49898 CDJQ32 127051599 IC50 = 66 nM T49898 CJ3M5I 134137436 Ki > 1000 nM T49898 CS4OW8 135400873 Ki = 35 nM T49898 CVJK60 135402835 IC50 = 260 nM T49898 COYA04 135402863 IC50 = 20 nM T49898 C9Y3WG 135404113 IC50 = 130 nM T49898 CDV48Y 135404796 IC50 = 200 nM T49898 CUY41E 135404846 IC50 = 45 nM T49898 CFOD89 135405216 IC50 = 77 nM T49898 CF39KX 135405229 IC50 = 150 nM T49898 CS7QH2 135405282 IC50 = 51 nM T49898 C82TVC 135409809 IC50 = 15 nM T49898 CH98WL 135418427 IC50 = 1700 nM T49898 CL46JK 135418490 IC50 = 10 nM T49898 C5ZQ0M 135421134 IC50 = 2300 nM T49898 CE8LA2 135421135 IC50 = 220 nM T49898 CWO64E 135421136 IC50 = 17 nM T49898 C3U0PF 135421137 IC50 = 7.1 nM T49898 C3A9UZ 135421138 IC50 = 130 nM T49898 C30VGC 135421139 IC50 = 2800 nM T49898 CRA56X 135421140 IC50 = 12 nM T49898 CT0D5M 135421141 IC50 = 19 nM T49898 CXZV53 135421142 IC50 = 16 nM T49898 CTRW73 135421143 IC50 = 740 nM T49898 CC84WV 135421144 IC50 = 29 nM T49898 C7TW3I 135421145 IC50 = 15 nM T49898 C9DUQ7 135421146 IC50 = 64 nM T49898 C3ERJ8 135421147 IC50 = 50 nM T49898 C13RGY 135421148 IC50 = 41 nM T49898 CEQ2X6 135421149 IC50 = 38 nM T49898 CE7LR5 135421150 IC50 = 12 nM T49898 C07BWX 135421151 IC50 = 72 nM T49898 CBUN39 135421152 IC50 = 41 nM T49898 CID92J 135421153 IC50 = 64 nM T49898 C29QXJ 135421154 IC50 = 14000 nM T49898 CFB7R0 135421155 IC50 = 52 nM T49898 CK7Y5X 135421156 IC50 = 910 nM T49898 C3R8LM 135421157 IC50 = 5500 nM T49898 C4SIP0 135421158 IC50 = 39 nM T49898 CMN0Q7 135421159 IC50 = 100 nM T49898 C6J9YR 135421160 IC50 = 170 nM T49898 CH50XP 135421161 IC50 = 1200 nM T49898 CY53SU 135421162 IC50 = 31 nM T49898 C3S7MX 135423008 IC50 > 1000 nM T49898 CEVL69 135423792 IC50 = 22000 nM T49898 CU60YC 135431661 IC50 = 3300 nM T49898 C4CXD1 135434964 IC50 = 1300 nM T49898 CFK9A4 135434965 IC50 = 300 nM T49898 C0ETV8 135434966 IC50 = 110 nM T49898 C9VM6D 135434967 IC50 = 46 nM T49898 CYBG82 135434968 IC50 = 37 nM T49898 C14BLP 135434969 IC50 = 19 nM T49898 CX16AQ 135434970 IC50 = 550 nM T49898 C3EU9C 135434971 IC50 = 41 nM T49898 C86TJA 135434972 IC50 = 290 nM T49898 C1QYE8 135434973 IC50 = 290 nM T49898 CZ63UC 135434975 IC50 = 150 nM T49898 CP95VZ 135434976 IC50 = 250 nM T49898 C52GQD 135434977 IC50 > 1000 nM T49898 C34YNR 135434978 IC50 = 290 nM T49898 CSLE24 135434979 IC50 = 95 nM T49898 CQT79I 135434980 IC50 = 210 nM T49898 CLP2K4 135434981 IC50 = 710 nM T49898 C8ZS4W 135434982 IC50 = 1400 nM T49898 C9XT7W 135434983 IC50 = 350 nM T49898 C6I1SH 135434984 IC50 = 170 nM T49898 C3S7WD 135434985 IC50 = 130 nM T49898 C45SHY 135434986 IC50 = 2.8 nM T49898 CSZ68Y 135434987 IC50 = 60 nM T49898 CN4MJ6 135434988 IC50 = 230 nM T49898 C2C3RF 135434989 IC50 = 74 nM T49898 CLYV03 135434990 IC50 = 60 nM T49898 CP8GA6 135434991 IC50 = 9.3 nM T49898 CN3A8I 135434992 IC50 = 520 nM T49898 CCP04J 135434993 IC50 = 660 nM T49898 C2VI7F 135434994 IC50 = 790 nM T49898 CBV6K4 135434995 IC50 > 1000 nM T49898 CY8W1P 135434996 IC50 > 10000 nM T49898 C1TN2K 135435000 IC50 = 250 nM T49898 CDM9R4 135435001 IC50 = 1700 nM T49898 C7M6WJ 135435002 IC50 = 87 nM T49898 CZSD45 135435003 IC50 = 120 nM T49898 CL0YS2 135435004 IC50 = 83 nM T49898 C64JZD 135435005 IC50 = 150 nM T49898 CGD0F2 135435006 IC50 = 43 nM T49898 CH41JZ 135435007 IC50 = 12 nM T49898 CBUR78 135435019 IC50 = 200 nM T49898 CCU3G9 135450829 IC50 = 45 nM T49898 C3IJ9V 135497787 IC50 = 8.5 nM T49898 C9YNE7 135497791 IC50 = 2.5 nM T49898 C8HO5W 135497794 IC50 = 110 nM T49898 CSP15M 135497800 IC50 > 1000 nM T49898 C0S3KJ 135497814 IC50 = 7.4 nM T49898 CBF73U 135497834 IC50 = 9 nM T49898 CEKY53 135497841 IC50 = 0.8 nM T49898 C7GKS9 135497849 IC50 = 0.7 nM T49898 C3WKV4 135497850 IC50 = 1.1 nM T49898 CTUB09 135497851 IC50 = 23 nM T49898 COH6V1 135497852 IC50 = 97 nM T49898 CU8T6K 135497853 IC50 = 41 nM T49898 CC58VR 135497854 IC50 = 5.6 nM T49898 C0ML5X 135497855 IC50 = 1.8 nM T49898 C1PJB2 135497865 IC50 = 13 nM T49898 C1V9AZ 135497869 IC50 = 39 nM T49898 CN2W4U 135497870 IC50 = 53 nM T49898 C03EJP 135497876 IC50 = 14 nM T49898 CR09SN 135497877 IC50 = 99 nM T49898 CU6T8C 135497878 IC50 = 1360 nM T49898 C45KEI 135497879 IC50 = 29 nM T49898 CK5G2W 135510524 IC50 = 3 nM T49898 CL5IR0 135512024 IC50 = 5 nM T49898 C8PRH9 135516527 IC50 = 290 nM T49898 CZY5G2 135566361 IC50 = 52 nM T49898 CM6C9G 135566570 IC50 = 94 nM T49898 C7PJ6X 135566704 IC50 > 30000 nM T49898 CRJ45X 135589980 IC50 > 50000 nM T49898 CFAD48 135611170 Ki = 20 nM T49898 C0J3BN 135678111 IC50 = 251 nM T49898 C95JVR 135744117 IC50 = 170 nM T49898 CYDM01 135891431 IC50 > 10000 nM T49898 CO6A1W 135950087 IC50 = 1580 nM T49898 C97HEY 136007770 IC50 = 31 nM T49898 C8BLU3 136007771 IC50 = 23 nM T49898 C3GVB5 136007772 IC50 = 31 nM T49898 C5NBU3 136025846 IC50 = 790 nM T49898 CEPW57 136025847 IC50 = 20 nM T49898 CT0N5U 136025985 IC50 = 7940 nM T49898 CFNZ81 136025987 IC50 = 2990 nM T49898 CJPT24 136025988 IC50 = 20 nM T49898 CWD1J4 136025989 IC50 = 280 nM T49898 CL1NP0 136026131 IC50 = 15 nM T49898 C26ESH 136060555 IC50 > 50000 nM T49898 CA0JB4 136068686 IC50 > 10000 nM T49898 C5BGL2 136068687 IC50 = 220 nM T49898 CXK3F8 136086909 IC50 = 19 nM T49898 CBC27R 136086910 IC50 = 45 nM T49898 CSM28V 136086911 IC50 = 340 nM T49898 C7FU8S 136086912 IC50 = 260 nM T49898 CWH74C 136086913 IC50 = 420 nM T49898 C60YSD 136086914 IC50 = 2240 nM T49898 CXV64Q 136086915 IC50 = 1000 nM T49898 C59GAN 136086916 IC50 = 10000 nM T49898 C20UHS 136086917 IC50 = 7500 nM T49898 C3X8QG 136086918 IC50 > 10000 nM T49898 C9KV0Y 136086919 IC50 > 10000 nM T49898 C1Y0PS 136118031 IC50 = 120 nM T49898 CA76XZ 136118032 IC50 = 10000 nM T49898 CVQ41X 136118033 IC50 = 540 nM T49898 CU5XR2 136118034 IC50 = 1280 nM T49898 C4G6PT 136118035 IC50 = 120 nM T49898 CRO6H1 136203706 IC50 = 2800 nM T49898 CAH27O 136219283 IC50 = 46.8 nM T49898 C61DOF 136274355 IC50 = 42 nM T49898 CH3M4B 137083628 IC50 > 30000 nM T49898 CJA07O 137083629 IC50 > 30000 nM T49898 C9F8PX 137083630 IC50 > 30000 nM T49898 C3DNL6 137349544 IC50 = 1520 nM T49898 CU9O3A 137628639 IC50 = 4.9 nM T49898 C25ERN 137631967 IC50 > 1000 nM T49898 C06JRX 137637094 IC50 > 1000 nM T49898 C1DK0P 137651391 IC50 > 1000 nM T49898 CV5H3Z 137657932 IC50 > 1000 nM T49898 C1LK7M 145975810 IC50 = 1413 nM T49898 CB2J4N 145989210 IC50 = 3 nM T49898 CR2GW6 145994117 IC50 = 1250 nM T49898 CZQM57 155554194 IC50 > 10000 nM T49898 CQ36LX 155555568 IC50 = 41 nM T49898 CAO81F 155563443 IC50 = 1900 nM T49898 CLXN40 155565350 IC50 = 578 nM T49898 C1NL5J 155566560 IC50 = 40 nM T49898 C8AOM4 11724428 IC50 = 6000 nM T49898 D00ERW 44444843 Ki > 8913 nM T49898 D00HVA 11624601 Ki > 8900 nM T49898 D00KDF 3387354 IC50 = 250 nM T49898 D03DZO 11715767 IC50 = 250 nM T49898 D04JIR 69689 IC50 > 350000 nM T49898 D04NGS 5330790 IC50 = 6 nM T49898 D04RBG 3536 IC50 = 100 nM T49898 D04TLB 135408762 IC50 = 6 nM T49898 D04YQF 763936 IC50 = 28000 nM T49898 D04ZWF 53396311 IC50 = 4000 nM T49898 D06BVH 18516979 IC50 > 10000 nM T49898 D07ADR 2422 IC50 = 2500 nM T49898 D07ADX 54764565 IC50 = 1125 nM T49898 D07OAT 456214 IC50 = 35000 nM T49898 D07SRX 9797919 IC50 > 10000 nM T49898 D08JML 10061827 IC50 = 13000 nM T49898 D08LYB 5166 IC50 > 50 nM T49898 D0BU6T 354471 IC50 = 54000 nM T49898 D0D2FC 2794188 IC50 = 110 nM T49898 D0D5ZL 369401 IC50 = 7000 nM T49898 D0D6DH 10125830 IC50 > 50000 nM T49898 D0E9DI 44430881 IC50 = 3500 nM T49898 D0EE6A 6398883 IC50 > 10000 nM T49898 D0EW9J 10389239 IC50 > 200000 nM T49898 D0FO2K 848641 IC50 > 200000 nM T49898 D0G2CT 3708 IC50 = 40 nM T49898 D0H3EV 5005498 IC50 = 35 nM T49898 D0L3FK 5289419 IC50 = 40 nM T49898 D0M5PI 10730551 IC50 = 3500 nM T49898 D0P2WA 6918386 IC50 = 330000 nM T49898 D0Q3KS 9957049 IC50 > 10000 nM T49898 D0Q3NG 11715520 Ki > 8900 nM T49898 D0QC0W 9914412 IC50 > 10000 nM T49898 D0R1FT 4564 Ki = 5000 nM T49898 D0S7IE 11658882 Ki > 8900 nM T49898 D0T4SJ 10356352 IC50 = 200 nM T49898 D0U8YN 398148 Ki = 2500 nM T49898 D0Y0ES 3707 IC50 = 180 nM T49898 D0Y5RO 4566 IC50 = 9.5 nM T49898 D0YE1X 9927943 IC50 > 10000 nM T49898 D0YM4A 22319604 IC50 = 100 nM T49898 D0YZ7H 9797370 IC50 > 100000 nM T49898 D0Z2CN 135418335 IC50 = 10000 nM T49898 D0Z8PT 54758482 IC50 > 10000 nM T43739 D03FLC 3878 IC50 = 96000 nM T43739 D0C7ET 11174599 IC50 > 30 nM T43739 D0X0RI 4178 IC50 = 56000 nM T43739 D04JZH 11659955 IC50 = 190 nM T43739 D04PER 49836093 IC50 = 4800 nM T43739 D0K9IF 71666749 IC50 = 15 nM T43739 D0O7QA 46840946 IC50 > 10000 nM T43739 D0OX9F 16046068 IC50 = 6000 nM T43739 CPN25U 998021 IC50 = 3000 nM T43739 CHW13G 16040159 IC50 = 19 nM T43739 CPCZ62 16040329 IC50 = 3 nM T43739 CTG41H 24778289 IC50 = 79 nM T43739 CF75YB 24857856 IC50 = 30 nM T43739 CBPY64 25008621 IC50 = 270 nM T43739 CTY4A0 25155168 IC50 = 920 nM T43739 CM8IJ3 25155169 IC50 = 750 nM T43739 CG0C3B 25155173 IC50 = 2400 nM T43739 CLZW63 25155700 IC50 = 670 nM T43739 CFB8E5 25159056 IC50 = 500 nM T43739 CP72MB 25159060 IC50 = 260 nM T43739 C9PUZ6 25159334 IC50 = 4900 nM T43739 CXWL81 44408928 Ki = 180 nM T43739 CIH69B 44445848 IC50 = 1000 nM T43739 C5C3YI 44447269 IC50 = 793 nM T43739 CF90DG 44447270 IC50 = 1458 nM T43739 C0WDU7 44447271 IC50 = 361 nM T43739 CUJ50E 44447273 IC50 = 230 nM T43739 C0HV4L 44447274 IC50 = 366 nM T43739 C4ZGH1 44447276 IC50 = 2975 nM T43739 C5MT0J 44447277 IC50 = 1782 nM T43739 C7PB9V 44447278 IC50 = 825 nM T43739 CIY3T7 44447280 IC50 = 880 nM T43739 CP7D3U 44447281 IC50 = 500 nM T43739 CC71MI 44447282 IC50 = 985 nM T43739 C0PT9W 44447287 IC50 = 685 nM T43739 C5NKU9 44447288 IC50 = 446 nM T43739 CX8GC7 44447290 IC50 = 295 nM T43739 CK6Q0S 44447291 IC50 = 806 nM T43739 CUW24D 44447292 IC50 = 1242 nM T43739 CYB0L8 44447295 IC50 = 1869 nM T43739 CHS74Q 44447296 IC50 = 446 nM T43739 CER76K 44585595 IC50 = 300 nM T43739 C40BIM 45139151 IC50 = 12400 nM T43739 CS5EJ1 46841648 IC50 > 10000 nM T43739 CRE97F 46841787 IC50 > 30000 nM T43739 CBXW47 50899559 IC50 = 14 nM T43739 C90UKY 50899643 IC50 = 23 nM T43739 CENW12 50925404 IC50 = 2000000 nM T43739 C63UYC 50925406 IC50 = 915 nM T43739 C06OXV 52920492 IC50 = 28000 nM T43739 C47GJP 52941142 IC50 = 2 nM T43739 C4J9VM 52942105 IC50 = 26 nM T43739 C6UO9M 52942117 IC50 = 9 nM T43739 C31XZV 52942252 IC50 = 140 nM T43739 C4VE8S 52942340 IC50 = 30 nM T43739 CVYW49 52943132 IC50 = 27 nM T43739 C3K0RO 52943146 IC50 = 6 nM T43739 CBR7A0 52943300 IC50 = 100 nM T43739 C9QAL2 52943533 IC50 = 8 nM T43739 C5BV9D 52944470 IC50 = 470 nM T43739 CM8SP7 52944476 IC50 = 8 nM T43739 CH54UW 52944738 IC50 = 2 nM T43739 CU5CL0 52945245 IC50 = 3 nM T43739 CTGW23 52945734 IC50 = 64 nM T43739 CDN9Y8 52945882 IC50 = 10 nM T43739 CI5BU7 52945890 IC50 = 7 nM T43739 CM2W7J 52945969 IC50 = 5 nM T43739 C7FMG4 52946920 IC50 = 2 nM T43739 C6U3TH 52946939 IC50 = 51 nM T43739 CEK18S 52947191 IC50 = 18 nM T43739 CJ6OG2 52947194 IC50 = 49 nM T43739 C4X3KP 52947201 IC50 = 1 nM T43739 CAQ8V0 52947207 IC50 = 150 nM T43739 C0NZ9X 52948309 IC50 = 8 nM T43739 CNA80Z 52948416 IC50 = 320 nM T43739 C6B0LV 52949221 IC50 = 19 nM T43739 CJFG89 52949235 IC50 = 6 nM T43739 CDP17N 52949384 IC50 = 280 nM T43739 CCI8B3 52949385 IC50 = 180 nM T43739 C5E6GD 52949400 IC50 = 21 nM T43739 CGQE06 52949417 IC50 = 780 nM T43739 CBC8U2 52949503 IC50 = 87 nM T43739 C1LBT3 52949586 IC50 = 99 nM T43739 C4QI5Y 52950155 IC50 = 37 nM T43739 CMS2F7 53239561 IC50 = 3770 nM T43739 CZMA05 53318633 IC50 = 299 nM T43739 CI3LN7 53318774 IC50 = 802 nM T43739 C8JF0H 53319960 IC50 = 203 nM T43739 C61MZW 53320375 IC50 = 554 nM T43739 CV9BR7 53321262 IC50 = 1513000 nM T43739 C73HYL 53321263 IC50 = 1181000 nM T43739 CM83SD 53326497 IC50 = 149 nM T43739 CR34CL 57582353 IC50 = 700 nM T43739 CETS76 59019389 IC50 > 1000 nM T43739 CZDW91 65458453 IC50 = 710 nM T43739 C9SEG5 65458673 IC50 > 1000 nM T43739 CC82DM 65459349 IC50 = 53 nM T43739 C0JSU4 65459575 IC50 = 1000 nM T43739 CWQZ40 67400361 IC50 = 417 nM T43739 CT1YQ7 68680505 IC50 = 24000 nM T43739 CMT89O 71111256 IC50 = 31000 nM T43739 C8RYJ4 71111280 IC50 = 3200 nM T43739 C09UZD 71111431 IC50 = 7000 nM T43739 C2MC6B 71522734 IC50 = 3850 nM T43739 CYPR67 71523540 IC50 = 190 nM T43739 CM1B0W 71523649 IC50 = 47 nM T43739 CG3L5O 71660502 IC50 = 10.5 nM T43739 CK68HF 71666608 IC50 = 18 nM T43739 CU0A9K 71666750 IC50 = 24 nM T43739 C9MUK3 71716856 IC50 > 3000 nM T43739 CUG2V3 71716866 IC50 > 10000 nM T43739 CLE3H9 71718687 IC50 = 680 nM T43739 CQ74UP 84626694 IC50 = 607 nM T43739 CTG76E 86687532 IC50 > 30000 nM T43739 C8UVE5 86699018 IC50 = 59 nM T43739 CLP5E2 86699068 IC50 = 227 nM T43739 C2SJ3Z 86699080 IC50 = 797 nM T43739 CRJ9F2 86699098 IC50 = 45 nM T43739 CN90UG 89738675 IC50 = 106 nM T43739 CSD20T 89845286 IC50 = 127 nM T43739 CQW6R8 89845320 IC50 = 130 nM T43739 CC3Y1N 89845361 IC50 = 31 nM T43739 C5O2KS 89845592 IC50 = 43 nM T43739 C9KV7L 117993993 IC50 = 15600 nM T43739 C7HJ6B 118126600 IC50 = 160 nM T43739 COCS31 118289757 IC50 = 579 nM T43739 C7AYV5 118540795 IC50 >= 10000 nM T43739 C3IDY0 122181194 IC50 > 32000 nM T43739 C0ZS7G 122181195 IC50 > 32000 nM T43739 CF97QP 122181196 IC50 > 32000 nM T43739 CG6U5Q 122181197 IC50 = 12000 nM T43739 CIHF48 122181198 IC50 > 32000 nM T43739 CC81BG 122181199 IC50 = 7400 nM T43739 C0SMG7 122181200 IC50 = 4000 nM T43739 CG1S2M 132519335 IC50 = 680 nM T43739 CO2SH1 132519336 IC50 = 1600 nM T43739 COP30C 132519337 IC50 = 390 nM T43739 CFB89A 137631484 IC50 > 1000 nM T43739 CUYN25 137631834 IC50 = 84 nM T43739 COQ47K 137631897 IC50 = 2200 nM T43739 CB4A0Y 137632255 IC50 = 2200 nM T43739 CNH92P 137634362 IC50 = 340 nM T43739 C86WPM 137638084 IC50 = 1600 nM T43739 CF29NZ 137639955 IC50 = 3200 nM T43739 CZSJ59 137640675 IC50 > 1000 nM T43739 CZS38R 137642807 IC50 = 230 nM T43739 C3K5IV 137645234 IC50 > 1000 nM T43739 CMG27C 137645959 IC50 = 3400 nM T43739 C7HVY4 137647174 IC50 = 260 nM T43739 CM9X7R 137652963 IC50 = 36 nM T43739 C0KU8R 137653454 IC50 = 620 nM T43739 C7HO5N 137655611 IC50 > 1000 nM T43739 C9JP7K 137657919 IC50 = 790 nM T43739 C65BRY 137658596 IC50 = 320 nM T43739 CN0HJ4 137659444 IC50 = 2600 nM T43739 CXM59Y 137660745 IC50 > 1000 nM T43739 CF6L8Q 145955101 IC50 = 509 nM T43739 CCTB54 145958837 IC50 > 1000 nM T43739 C38DYW 145959291 IC50 > 1000 nM T43739 CZN0U6 145982478 IC50 = 15100 nM T43739 C8Q2EG 145988110 IC50 = 11300 nM T43739 C3LJ1I 155515503 IC50 > 1000 nM T43739 C5Y9SK 155516393 IC50 = 593 nM T43739 C8F2NE 155519037 IC50 = 534 nM T43739 CY1NX3 155525154 IC50 > 1000 nM T43739 CJ21QH 155525808 IC50 = 43 nM T43739 C86XSP 155527173 IC50 = 728 nM T43739 CCH9L7 155540658 IC50 = 2 nM T43739 CZ04LB 155542770 IC50 = 95 nM T43739 CXK70M 155546234 IC50 = 998 nM T43739 CZ5G4W 155547025 IC50 = 708 nM T43739 CAPU04 155553341 IC50 = 65 nM T43739 CW0C9F 155554474 IC50 = 742 nM T43739 C0AJ7O 155560387 IC50 > 1000 nM T43739 CMLC50 155566454 IC50 = 2567 nM T43739 CE3H4Z 155567528 IC50 = 50000 nM T43739 C4Z3TO 155567878 IC50 > 1000 nM T43739 CU6NG3 155568346 IC50 > 1000 nM T43739 D01AGR 24857857 IC50 = 280 nM T43739 D02CQN 52945923 IC50 = 2 nM T43739 D0F5WY 44435593 IC50 = 9000 nM T43739 D0FF6S 16038374 IC50 = 8 nM T43739 D0O0JO 52948346 IC50 = 4 nM T43739 D0P8TL 56947150 IC50 > 10000 nM T43739 D0W2BP 46032908 IC50 = 22 nM T61317 D04AIT 5280445 Ki = 800 nM T61317 D0K8KX 5280343 IC50 = 5400 nM T61317 D0U2BH 65064 IC50 = 0.32 ug.mL-1 T61317 CNIW58 107905 IC50 = 1000 nM T61317 CDZ65K 199472 IC50 = 1100 nM T61317 CN7AQ6 15958429 IC50 > 100 ug.mL-1 T61317 CZR73C 16072317 IC50 > 100 ug.mL-1 T61317 C20YLR 22600366 IC50 = 3.5 ug.mL-1 T61317 C6XHE9 49770727 IC50 > 100 ug.mL-1 T61317 D01UYI 5281607 IC50 = 10000 nM T61317 D02TVS 985 IC50 > 100 ug.mL-1 T61317 D06NRZ 188323 IC50 = 70000 nM T61317 D07YDN 5281654 IC50 = 8300 nM T61317 D0G3TK 5280863 IC50 = 4000 nM T61317 D0MF5Y 5281614 IC50 = 4100 nM T61317 D0NJ4H 5281670 IC50 = 2300 nM T61317 D0RB1V 6419835 IC50 = 1000 nM T61317 D0T3PW 5281672 IC50 = 14000 nM T61317 D0Y7HG 5281616 IC50 = 100000 nM T98397 D01KKQ 135400182 IC50 = 290 nM T98397 D0SV8E 126941 Ki = 600 nM T98397 D0Y4GO 135410875 Ki = 1.3 nM T98397 D0Z0DW 135398658 Ki = 40000 nM T98397 D06WQT 135400184 Ki = 15 nM T98397 D03FDT 4764 Ki = 1200 nM T98397 D06YIB 135436405 IC50 > 1000000 nM T98397 D0C4YA 3047716 Ki = 2 nM T98397 D0TP9A 135528987 IC50 = 156 nM T98397 C7OTP8 3439 IC50 > 200000 nM T98397 C5VX1C 6693 Ki = 2000 nM T98397 CLD7W2 18194 Ki > 206000 nM T98397 CLMB45 77672 Ki = 7300 nM T98397 C5L9YZ 78907 Ki = 4200 nM T98397 CH3MC1 80990 Ki > 160000 nM T98397 CF6GB0 96894 Ki > 309000 nM T98397 CU51YB 104070 Ki > 824000 nM T98397 CGOP98 132151 Ki = 1600 nM T98397 CZA4M3 158351 IC50 > 200000 nM T98397 CCX59F 163544 Ki = 2000 nM T98397 CTSM43 174519 Ki = 4.77 nM T98397 CL5Y6C 223824 Ki = 47000 nM T98397 C4CPL5 290624 Ki > 309000 nM T98397 CXA5L9 305193 Ki = 12000 nM T98397 CM8L9N 361689 IC50 = 619000 nM T98397 C8WO4J 403898 Ki > 402000 nM T98397 CTO2D8 404585 Ki = 51000 nM T98397 C2IZ4Q 405137 Ki = 6000 nM T98397 C0MKV6 405140 Ki = 25000 nM T98397 CIZ2O5 405953 Ki = 34000 nM T98397 CDC2L4 406510 Ki = 5000 nM T98397 C65ECP 448780 Ki = 30000 nM T98397 CF1M8Q 468708 IC50 > 200000 nM T98397 CRB65P 481401 IC50 > 16000 nM T98397 CZQ3G2 484977 Ki > 120000 nM T98397 CHEO87 604195 Ki = 3100 nM T98397 C5KGM0 899290 Ki = 10000 nM T98397 C61CNA 2781167 Ki > 474000 nM T98397 CDQU17 3513688 Ki > 98000 nM T98397 C3VU7M 3604775 Ki = 2000 nM T98397 CC26SD 4149717 Ki = 3100 nM T98397 C56EON 4530276 Ki > 309000 nM T98397 CHGZ97 5288461 IC50 = 1000 nM T98397 CZ5D6N 6443208 Ki = 8600 nM T98397 CVD9P3 6876724 IC50 = 112000 nM T98397 C02TVS 9845472 Ki = 770 nM T98397 CC36EP 9889551 IC50 = 63000 nM T98397 C5VZN4 9911146 IC50 > 360000 nM T98397 C3GI6F 9931657 Ki > 5000 nM T98397 CL0P6O 9932276 IC50 = 220000 nM T98397 CDSX76 9947879 Ki = 17 nM T98397 CIDQ05 9952879 Ki > 5000 nM T98397 C1VC0I 9954209 Ki = 64 nM T98397 C0NZC8 9994347 Ki = 15 nM T98397 C5R4GN 10358404 Ki = 25 nM T98397 C7Q1OZ 10363363 Ki = 52 nM T98397 CTB38W 10380195 Ki = 6 nM T98397 C02XZU 10402662 Ki = 14 nM T98397 CHO93B 10402730 Ki = 10 nM T98397 C7KXJ2 10404647 IC50 = 110 nM T98397 CTX6H7 10433577 IC50 = 540 nM T98397 CG9TR7 10450905 Ki = 45 nM T98397 CZD4B0 10456691 IC50 > 18000 nM T98397 CHM3X4 10478775 Ki > 132000 nM T98397 CC5O2D 10520145 Ki = 10300 nM T98397 C9LPA1 10993870 IC50 = 80000 nM T98397 CT6N3U 11117688 Ki = 33000 nM T98397 C1VO8F 11723304 Ki = 4 nM T98397 C0Z7NG 11723407 Ki = 18 nM T98397 CQ4H5E 11744008 IC50 > 18000 nM T98397 CR9GN2 11826533 IC50 = 9000 nM T98397 C0L5BK 12680923 Ki > 412000 nM T98397 C4L3SC 14542115 IC50 = 11300 nM T98397 C4DHV7 15131016 Ki = 13.1 nM T98397 CZRO46 15131017 Ki = 20 nM T98397 CH23LW 15131018 Ki = 24 nM T98397 CW9E1R 15131019 Ki = 38 nM T98397 CL8M2A 15131020 Ki = 6 nM T98397 C59PXH 15131021 Ki = 7700 nM T98397 C8I9DO 15131023 Ki = 4200 nM T98397 CB2K3X 15131024 Ki = 770 nM T98397 C0GCS5 15131026 Ki = 51 nM T98397 CO97SV 15131027 Ki = 440 nM T98397 CGJ84O 15131028 Ki = 480 nM T98397 C84ABT 15131041 Ki = 230 nM T98397 CKD51Y 15169667 Ki = 31 nM T98397 CHF58K 15169677 Ki = 840 nM T98397 CWKX69 16086910 Ki > 132000 nM T98397 C6V7GN 16086911 Ki = 400 nM T98397 C3X9DE 16086912 Ki > 245000 nM T98397 C9KZ4H 16086913 Ki > 132000 nM T98397 CTK25X 16086914 Ki > 245000 nM T98397 CD59VR 16086916 Ki = 34000 nM T98397 C6UX1P 16086917 Ki > 132000 nM T98397 CRWB95 16086918 Ki > 245000 nM T98397 C0RE7Z 16086919 Ki > 245000 nM T98397 CUSF67 23648073 Ki > 132000 nM T98397 CI2F9K 23648074 Ki = 5700 nM T98397 C4SXQ7 23648075 Ki = 4700 nM T98397 CDUX91 23648076 Ki = 3200 nM T98397 C4S9RX 24202946 Ki = 3560 nM T98397 C6H1RM 24202947 Ki = 2380 nM T98397 C7AXQ6 24203165 Ki = 510 nM T98397 C58NDL 24203444 Ki = 900 nM T98397 C5S8PW 24204221 Ki = 270 nM T98397 CPG6Z7 24796532 Ki = 15000 nM T98397 C7H5WQ 24796533 Ki = 21000 nM T98397 C9I5ST 24796666 Ki = 700 nM T98397 CBD1J8 24796667 Ki = 14000 nM T98397 C3C8LF 24796668 Ki = 36000 nM T98397 CL7KN4 24950538 IC50 > 22000 nM T98397 C2C4FZ 24950539 IC50 > 24000 nM T98397 C9LY5G 24950540 IC50 > 14000 nM T98397 CPEF92 24950541 IC50 > 13000 nM T98397 CD8QM2 24950542 IC50 > 12000 nM T98397 CX5Q0K 24950543 IC50 > 11000 nM T98397 CH9A4V 24950693 IC50 > 12000 nM T98397 CG6A8V 24950694 IC50 > 12000 nM T98397 C6F2CR 24950695 IC50 > 22000 nM T98397 CX1AR8 24950696 IC50 > 13000 nM T98397 C1PHA0 24950697 IC50 > 27000 nM T98397 CG2B8O 24950698 IC50 > 25000 nM T98397 CX97IY 24950699 IC50 > 23000 nM T98397 C32OJF 24950851 IC50 > 23000 nM T98397 CCY8U4 24950852 IC50 > 12000 nM T98397 C17DAP 24950853 IC50 > 24000 nM T98397 CPDN34 24950854 IC50 > 23000 nM T98397 C6W1TN 25107577 IC50 = 1200 nM T98397 CHU9G1 25107640 IC50 = 260 nM T98397 C5WV3Q 25107642 IC50 = 1000 nM T98397 C2FU7W 25107643 IC50 = 280 nM T98397 C5EP2L 25107644 IC50 = 110 nM T98397 C3YT9V 25107645 IC50 = 120 nM T98397 CQV0S4 25107646 IC50 = 1100 nM T98397 CT3CA2 25134257 Ki = 81000 nM T98397 COB9G8 25181586 IC50 = 540 nM T98397 C8IJB9 25218207 IC50 = 390 nM T98397 CI0BF4 44201386 IC50 = 54 nM T98397 CZ6DE0 44221143 IC50 = 750 nM T98397 CL8B5Q 44221144 IC50 = 4600 nM T98397 CSJ28V 44221145 IC50 = 690 nM T98397 COT01Q 44221146 IC50 = 1300 nM T98397 CS14YU 44221147 IC50 = 380 nM T98397 CA64NZ 44221340 IC50 = 1100 nM T98397 CK5OL1 44221343 IC50 = 5600 nM T98397 CW0IM7 44221344 IC50 = 220 nM T98397 C0QZ7V 44221345 IC50 = 230 nM T98397 C74PHB 44221346 IC50 = 2300 nM T98397 CW39YO 44221347 IC50 = 280 nM T98397 CBHT60 44221538 IC50 = 390 nM T98397 CN5QV6 44221539 IC50 = 1200 nM T98397 C2DQ9E 44300934 IC50 = 220000 nM T98397 CN9U6W 44300964 IC50 > 360000 nM T98397 CEV8X6 44300967 IC50 = 220000 nM T98397 CKN1S7 44325462 IC50 = 430 nM T98397 CU78HI 44325575 IC50 = 740 nM T98397 CU98BO 44325666 IC50 = 24000 nM T98397 C04VSI 44327287 IC50 = 3100 nM T98397 CN4Y5S 44373841 IC50 = 1260 nM T98397 C2Z5JN 44373979 IC50 = 20000 nM T98397 C5F0ZB 44378252 Ki > 5000 nM T98397 CZ7Y4L 44378321 Ki > 5000 nM T98397 C3W2YH 44378322 Ki > 5000 nM T98397 CQY9S6 44381789 Ki = 11 nM T98397 CUWB37 44388290 Ki = 11 nM T98397 CD50BE 44388299 Ki = 4.1 nM T98397 CT57RK 44388300 Ki = 8.5 nM T98397 C70CFI 44388301 Ki = 1.5 nM T98397 CE84PW 44388306 Ki = 13 nM T98397 C9DU4Y 44448712 Ki = 432800 nM T98397 CX5YK8 44567483 Ki = 16000 nM T98397 CN76FA 44568860 IC50 = 40 nM T98397 C7Q5KD 44788406 Ki = 300 nM T98397 CST4J2 44788425 Ki = 1100 nM T98397 CSW75Q 44788432 Ki = 500 nM T98397 C1YAE7 46231368 IC50 = 5400 nM T98397 C1PJ2K 46231369 IC50 > 200000 nM T98397 CV38CS 46231370 IC50 > 200000 nM T98397 C5WM1J 46231371 IC50 > 200000 nM T98397 C5D7UV 46231372 IC50 > 200000 nM T98397 C9OER4 46231373 IC50 > 200000 nM T98397 CW0UO4 46231409 IC50 > 200000 nM T98397 C7OG0U 46231410 IC50 > 200000 nM T98397 CU5T7G 46231411 IC50 > 200000 nM T98397 COML63 46231412 IC50 > 200000 nM T98397 CK21OD 46231413 IC50 > 200000 nM T98397 C7Y5MX 46231414 IC50 > 200000 nM T98397 CQ76PW 46840167 Ki = 43000 nM T98397 CO8X1S 49796223 Ki = 3000 nM T98397 C3NTG6 52911805 IC50 = 3900 nM T98397 CD6T0F 52911806 IC50 = 3600 nM T98397 C3H1RO 52911859 IC50 = 3200 nM T98397 CP85JZ 52911912 IC50 = 2100 nM T98397 CJA45X 52914860 IC50 = 68 nM T98397 CV21AI 52914861 IC50 = 34 nM T98397 CE02NU 52943039 IC50 > 360000 nM T98397 C7FZ3B 53392517 Ki = 48000 nM T98397 CC18TD 53392519 Ki = 206000 nM T98397 C07YBI 53392520 Ki = 21000 nM T98397 CT9BP0 53392605 Ki = 60000 nM T98397 C2LK8T 53392607 Ki = 30000 nM T98397 CJU65L 53964379 Ki = 60 nM T98397 COQC79 54678804 IC50 = 71000 nM T98397 CUPO65 56666113 IC50 = 260 nM T98397 C6RCQ7 56676341 IC50 = 800 nM T98397 CBOX49 59608000 Ki = 64000 nM T98397 C08ZJI 71520245 Ki = 17300 nM T98397 CIQ70J 71520246 Ki = 25400 nM T98397 CE83DS 71520247 Ki = 1300 nM T98397 C8MD9O 71520248 Ki = 12300 nM T98397 CDF29U 71520249 Ki = 1200 nM T98397 C34EBQ 71520250 Ki = 13800 nM T98397 C9IC0F 71520251 Ki = 800 nM T98397 C9SU7T 71520360 Ki > 411000 nM T98397 C2UCE5 71520361 Ki = 300 nM T98397 CLJ2Q5 71520362 Ki = 16200 nM T98397 CSWH97 71520363 Ki = 5000 nM T98397 CWF43X 71520364 Ki = 57200 nM T98397 CWX6T2 71520365 Ki = 600 nM T98397 C3B4HF 71520366 Ki > 616000 nM T98397 CHS24Z 71520480 Ki = 800 nM T98397 C76MAS 71520481 Ki > 206000 nM T98397 C1SP2K 71520482 Ki > 826000 nM T98397 C9M2JK 71520483 Ki = 25900 nM T98397 C5N4XG 71521660 Ki = 2300 nM T98397 CMQY40 71521740 Ki > 823000 nM T98397 CIZ23J 71521741 Ki = 1300 nM T98397 C8PK4V 71521742 Ki > 206000 nM T98397 C4YZ9L 71521743 Ki = 44600 nM T98397 CPJ46E 71521744 Ki = 900 nM T98397 C65NLD 71584213 IC50 = 620 nM T98397 C28AET 71584343 IC50 = 1600 nM T98397 C8F1HW 71584348 IC50 = 890 nM T98397 CMSJ92 71584467 IC50 = 1200 nM T98397 CZV86E 71584469 IC50 = 920 nM T98397 CMW7B2 71584470 IC50 = 2200 nM T98397 C6HEK1 71584472 IC50 = 1700 nM T98397 C26DSY 71768362 Ki = 35000 nM T98397 C54ADX 72737236 Ki = 7000 nM T98397 CAHW96 72737238 Ki = 60000 nM T98397 C5KH0G 72737239 Ki = 8000 nM T98397 CI36PZ 72737240 Ki = 28000 nM T98397 C0HSC8 73346520 Ki = 3650 nM T98397 C8SD9P 73346521 Ki = 6220 nM T98397 CGZ6Y8 73346522 Ki = 3730 nM T98397 C43IPQ 73348006 Ki = 340 nM T98397 CS9C0W 73351108 Ki = 19270 nM T98397 C27JUH 73352576 Ki = 11340 nM T98397 CVP03Z 73352577 Ki = 1140 nM T98397 CDAB86 73354065 Ki = 5600 nM T98397 CK3Z8U 73354066 Ki = 1360 nM T98397 C92DXZ 73354067 Ki = 4060 nM T98397 CCI18Y 73355591 Ki = 5090 nM T98397 CRX8A0 73355592 Ki = 10910 nM T98397 CTXE70 76314510 Ki = 26000 nM T98397 C9MVU4 76318086 IC50 = 300000 nM T98397 C60EOK 90663731 Ki = 58700 nM T98397 C5YSP3 90663787 Ki = 6800 nM T98397 C8OTU1 90663788 Ki = 5600 nM T98397 C61XNE 90663789 Ki = 39400 nM T98397 CDBA59 90663790 Ki = 15400 nM T98397 CBC85O 90663791 Ki = 29400 nM T98397 CQ6W3F 90663792 Ki = 134100 nM T98397 C34DLF 90663793 Ki = 66300 nM T98397 CS6JB4 90663794 Ki = 114200 nM T98397 C4HZ6K 90663795 Ki = 35000 nM T98397 CB64IZ 90663796 Ki = 119400 nM T98397 CCPZ32 90663797 Ki = 21700 nM T98397 CH7SD4 90663798 Ki = 102500 nM T98397 C5FJR8 118725249 Ki = 30 nM T98397 C8G7BW 118730356 Ki = 60000 nM T98397 CMQ9I8 118730357 IC50 = 52000 nM T98397 C78DHJ 118730358 IC50 = 56000 nM T98397 CX48ZK 118730359 IC50 = 88000 nM T98397 CZM06X 118730360 IC50 = 57000 nM T98397 CLFB23 118730361 IC50 = 300000 nM T98397 C1QVE3 121378588 IC50 > 100000 nM T98397 CSY29D 135399661 IC50 = 2700 nM T98397 CCT84X 135399760 IC50 = 100000 nM T98397 C68HXG 135399909 IC50 = 26000 nM T98397 C92RHD 135400923 Ki > 10000 nM T98397 CQ4F8Y 135402053 Ki = 4.5 nM T98397 C6AY2U 135403832 Ki = 0.09 nM T98397 C0LTC1 135404992 IC50 = 42 nM T98397 CD46CR 135405044 Ki = 1.2 nM T98397 C9EA3J 135407589 IC50 > 100000 nM T98397 C64LOS 135410241 Ki > 100000 nM T98397 C8IGV6 135410337 Ki = 39 nM T98397 CH37GZ 135411257 Ki = 2200 nM T98397 CZR7Y2 135412767 Ki = 8800 nM T98397 CO27TG 135413520 IC50 = 2040 nM T98397 C3MHI2 135427303 IC50 = 1800 nM T98397 CBT64V 135427959 IC50 = 1100 nM T98397 CL94UK 135427960 IC50 = 1000 nM T98397 C13MON 135428091 Ki = 310 nM T98397 C42MKL 135430799 Ki = 1.1 nM T98397 CZ5TY0 135430807 Ki = 0.09 nM T98397 CT16LV 135430817 IC50 = 156 nM T98397 CSNH87 135431649 IC50 = 54 nM T98397 C4T2WN 135433918 Ki = 58 nM T98397 CW3B5U 135434845 Ki = 1000 nM T98397 CH07YM 135438181 Ki = 120000 nM T98397 CZY6W8 135442802 Ki = 270 nM T98397 C5SL9R 135444566 Ki = 37 nM T98397 CZ65LS 135449121 Ki = 87 nM T98397 CRL53F 135453212 IC50 = 16000 nM T98397 C4RT3F 135453938 Ki = 58 nM T98397 C1M4UI 135455959 Ki = 12 nM T98397 C3X1SW 135456000 IC50 = 180 nM T98397 CFD9Y4 135456707 IC50 = 30000 nM T98397 CQ8B0H 135457333 Ki = 65 nM T98397 CHW12U 135461208 IC50 = 5600 nM T98397 CCS4A0 135461759 IC50 = 5300 nM T98397 C3W6CJ 135462247 IC50 = 2400 nM T98397 CEZI23 135464133 Ki = 14 nM T98397 CA9VC4 135464136 Ki = 30 nM T98397 CA2L6T 135464152 Ki = 32 nM T98397 CGSA26 135464205 Ki = 70 nM T98397 CNTX16 135469124 Ki = 22 nM T98397 CIB91S 135474272 Ki = 310 nM T98397 CK0LS8 135474356 Ki = 56 nM T98397 C8OYD4 135474773 Ki = 4 nM T98397 CF51JL 135475906 IC50 = 230 nM T98397 CH6L8Y 135485660 IC50 = 156 nM T98397 CJ5F0E 135487332 IC50 = 5600 nM T98397 C2IY5A 135487364 IC50 = 210 nM T98397 C7BQ1O 135487985 IC50 = 90 nM T98397 C0PD9J 135488011 Ki = 21 nM T98397 CI1AR4 135488050 Ki = 2.5 nM T98397 CQ5VE0 135491882 IC50 = 2600 nM T98397 C76QDH 135492362 Ki = 960 nM T98397 CP3Y7S 135492393 Ki = 11 nM T98397 CJV87K 135501139 Ki = 37 nM T98397 CD40CJ 135502983 IC50 = 220 nM T98397 CD32BW 135503936 Ki = 61 nM T98397 CVXL95 135511146 IC50 > 25000 nM T98397 C98GZD 135511915 IC50 = 130 nM T98397 CQ1HE7 135516687 IC50 = 340 nM T98397 CFH82R 135516724 IC50 = 1400 nM T98397 CDZ3E4 135516742 Ki = 200 nM T98397 CRQB90 135516748 Ki = 18 nM T98397 C6DVH0 135517330 Ki = 24 nM T98397 CC1XK2 135517445 Ki = 76 nM T98397 C8ZKI6 135524511 Ki = 260 nM T98397 C5MQU4 135525421 IC50 = 416.87 nM T98397 CZW50S 135527705 IC50 = 5000 nM T98397 C2XWJ5 135529900 Ki = 390 nM T98397 C4TM6O 135530074 IC50 = 240 nM T98397 CLB45I 135543610 IC50 = 130 nM T98397 CR1B7N 135543794 Ki = 27 nM T98397 CK4FS8 135543796 Ki = 26 nM T98397 CP75MF 135543822 IC50 = 19.95 nM T98397 CV7HQ6 135545795 IC50 = 4600 nM T98397 C8N5QD 135545810 IC50 > 17000 nM T98397 C9K8DE 135545856 IC50 = 51 nM T98397 CP3L1K 135545871 Ki = 0.44 nM T98397 CB2MI3 135564900 Ki = 69 nM T98397 CZ6Q7M 135566834 Ki = 55.7 nM T98397 CV6UW9 135566835 Ki = 378 nM T98397 C9Z4ES 135567027 IC50 > 17000 nM T98397 C6OW4E 135588787 IC50 = 5700 nM T98397 CEOY84 135600305 IC50 = 2700 nM T98397 C2EF4X 135622210 IC50 = 600 nM T98397 CFEH39 135625306 IC50 = 5500 nM T98397 CLCR96 135625340 IC50 = 4466.84 nM T98397 C74RXK 135625341 IC50 = 478.63 nM T98397 C7JHN2 135659594 Ki = 7370 nM T98397 CXZD49 135718456 IC50 = 5754.4 nM T98397 CNF8T7 135722138 IC50 = 141.25 nM T98397 C8T4XL 135722139 IC50 = 97.72 nM T98397 CN21RT 135722140 IC50 = 67.61 nM T98397 C2V7BF 135722141 IC50 = 239.88 nM T98397 CDT76J 135722142 IC50 = 44.67 nM T98397 C32ESM 135722144 IC50 = 302 nM T98397 CX06FR 135722145 IC50 = 371.54 nM T98397 CJL6U7 135722146 IC50 = 169.82 nM T98397 C9CT5W 135722147 IC50 = 144.54 nM T98397 C45UFQ 135722148 IC50 = 239.88 nM T98397 CA9U4J 135722156 IC50 = 89.13 nM T98397 C06IDH 135746097 Ki = 8.5 nM T98397 C2SB5J 135746748 Ki = 93000 nM T98397 CGLI18 135749904 IC50 = 46 nM T98397 CQ49YZ 135749905 IC50 = 20000 nM T98397 CBUS79 135749906 IC50 = 2300 nM T98397 C2HZK8 135749907 IC50 = 3700 nM T98397 CD48XU 135749908 IC50 = 2900 nM T98397 C9NZA4 135749909 IC50 = 1300 nM T98397 C0ME1H 135749910 IC50 = 1400 nM T98397 CMVH39 135749911 IC50 = 1500 nM T98397 CR4DU1 135749912 IC50 = 1300 nM T98397 C1H6ZF 135749913 IC50 > 26000 nM T98397 CR5NK7 135749914 IC50 = 10000 nM T98397 C1LV7B 135749915 IC50 = 5400 nM T98397 CCJ68D 135777639 IC50 = 55000 nM T98397 COV1E6 135777640 IC50 = 290 nM T98397 CQF8P5 135800109 IC50 > 17000 nM T98397 C08PIA 135813030 IC50 = 575.44 nM T98397 C9TWU2 135813031 IC50 = 263.03 nM T98397 CLH29C 135813032 IC50 = 758.58 nM T98397 C2P9FE 135813745 IC50 = 3100 nM T98397 CM0LN8 135817419 IC50 = 1.2 nM T98397 CB6ZP7 135838100 IC50 = 83600 nM T98397 CFP97G 135838102 IC50 = 230 nM T98397 CH0NX8 135838103 IC50 = 7160 nM T98397 CXT0E4 135838108 IC50 = 51000 nM T98397 CGT4X9 135838109 IC50 = 8400 nM T98397 CDSN50 135838114 IC50 = 6000 nM T98397 C4QYS5 135838116 IC50 = 145500 nM T98397 CE4V6Y 135838117 IC50 = 1150 nM T98397 C5AU6F 135838119 IC50 = 156000 nM T98397 CHNY32 135838121 IC50 = 120 nM T98397 C1I8LH 135838122 IC50 = 35600 nM T98397 C0SDR8 135838124 IC50 = 343 nM T98397 CGLZ87 135838125 IC50 = 360 nM T98397 CM3KJ7 135838126 IC50 = 3000 nM T98397 C7DTZ0 135838128 IC50 = 19000 nM T98397 CTD98I 135838129 IC50 = 13490 nM T98397 CEF9B1 135838130 IC50 = 710 nM T98397 C91WNF 135838132 IC50 = 26000 nM T98397 CA5ZU1 135838133 IC50 = 192800 nM T98397 CO83HS 135838134 IC50 = 1800 nM T98397 CK1U4F 135838135 IC50 = 1550 nM T98397 CJ4T9E 135838138 IC50 = 6500 nM T98397 CU29JG 135838139 IC50 = 480 nM T98397 C4LAP0 135838141 IC50 = 3900 nM T98397 CGL7Z0 135838142 IC50 = 16800 nM T98397 C9VK1A 135838145 IC50 = 6900 nM T98397 CKU2M1 135838148 IC50 = 3600 nM T98397 CE56FY 135838152 IC50 = 146000 nM T98397 CEN64U 135838153 IC50 = 4200 nM T98397 CB1RV4 135838155 IC50 = 290 nM T98397 CW1N3C 135838157 IC50 = 25000 nM T98397 CL19UJ 135838158 IC50 = 1600 nM T98397 CV6HL2 135838161 IC50 = 540 nM T98397 CCEA56 135838162 IC50 = 15200 nM T98397 CZ6QT7 135838168 IC50 = 27000 nM T98397 CKIW97 135838170 IC50 = 15000 nM T98397 CIL06X 135838171 IC50 = 7500 nM T98397 C86TUC 135838172 IC50 = 43900 nM T98397 C97BTY 135838173 IC50 = 17000 nM T98397 CBZ89A 135838174 IC50 = 24000 nM T98397 C3BC8N 135838175 IC50 = 630 nM T98397 CQD0K5 135838178 IC50 = 154000 nM T98397 C2VJ3Q 135838179 IC50 = 1000 nM T98397 C5YAI6 135838181 IC50 = 58900 nM T98397 C9X4QH 135838182 IC50 = 7500 nM T98397 CT1Z4N 135838183 Ki = 9000 nM T98397 C3T6RD 135838184 IC50 = 8600 nM T98397 C80OCL 135838187 IC50 = 520 nM T98397 C8ST9L 135838189 IC50 = 20 nM T98397 CJ5G8F 135838190 IC50 = 1600 nM T98397 CW09PU 135838191 IC50 = 32100 nM T98397 CLP64G 135838196 IC50 = 220000 nM T98397 CWU5P0 135838197 IC50 = 52500 nM T98397 CPB2W1 135838199 IC50 = 102 nM T98397 CFS49O 135838200 IC50 = 21000 nM T98397 C24CLA 135838201 IC50 = 44000 nM T98397 CTD12N 135838205 IC50 = 490 nM T98397 CA9MF3 135838207 IC50 = 107000 nM T98397 CR2E0S 135838209 IC50 = 73000 nM T98397 CF3P8N 135838210 IC50 = 79000 nM T98397 C7KH0P 135838211 IC50 = 2600 nM T98397 C2P8RA 135838213 IC50 = 3280 nM T98397 C9E8SH 135838214 IC50 = 2800 nM T98397 C2X3FW 135838216 IC50 = 22 nM T98397 C3S0VA 135838217 IC50 = 500 nM T98397 CU14CM 135838218 IC50 = 73800 nM T98397 CY1CV8 135838222 IC50 = 34000 nM T98397 CMRW42 135838223 IC50 = 8900 nM T98397 C84BXI 135838225 IC50 = 34500 nM T98397 C7HV0N 135838226 IC50 = 7800 nM T98397 CL47CY 135838227 IC50 = 25 nM T98397 CZ3S0O 135838229 IC50 = 157 nM T98397 CLN8J7 135838230 IC50 = 440 nM T98397 C6AB5J 135838231 IC50 = 28700 nM T98397 CM3US1 135838232 IC50 = 1980 nM T98397 CQ5L6G 135838233 IC50 = 460 nM T98397 C2NIC1 135838235 IC50 = 1310 nM T98397 C4WD0G 135838236 IC50 = 370 nM T98397 CE76RM 135838238 IC50 = 720 nM T98397 CHG5I6 135838239 IC50 = 552000 nM T98397 CV1QZ9 135838240 IC50 = 45400 nM T98397 C29WFU 135838242 IC50 = 8800 nM T98397 C5I8AD 135838243 IC50 = 40400 nM T98397 C57GYF 135838244 IC50 = 340 nM T98397 C3SDM6 135838245 IC50 = 3120 nM T98397 CE6L1M 135838246 IC50 = 154000 nM T98397 CL60XY 135838248 IC50 = 15600 nM T98397 CDLS80 135838249 IC50 = 22000 nM T98397 CTG51U 135887103 IC50 = 300000 nM T98397 CY5H4A 135887105 IC50 = 55000 nM T98397 CHT2O4 135887106 IC50 = 4200000 nM T98397 CWL71S 135887124 IC50 = 470000 nM T98397 CNKW46 135887125 IC50 = 2100000 nM T98397 CH1W2S 135887126 IC50 = 7100 nM T98397 C6U0PF 135887127 IC50 = 480 nM T98397 COA6S0 135887128 IC50 = 28800 nM T98397 CFIG79 135887147 IC50 > 100000 nM T98397 CDA05G 135887148 IC50 > 100000 nM T98397 C9TL7I 135958359 Ki = 2 nM T98397 CZB8O6 135960753 IC50 = 4600 nM T98397 COD5U9 135964377 IC50 = 2300 nM T98397 C43TOZ 135964378 IC50 = 460 nM T98397 C6B8AD 135964380 IC50 = 1200 nM T98397 C4IL6J 135964387 IC50 = 2800 nM T98397 CZ6C4R 135964391 IC50 = 800 nM T98397 CUOV62 135964392 IC50 = 280 nM T98397 CG23QU 135964393 IC50 = 1400 nM T98397 CR5EG8 135964397 IC50 = 460 nM T98397 C0T2QO 135964404 IC50 = 2700 nM T98397 CD8WY9 135964405 IC50 > 21000 nM T98397 CRXF18 135964411 IC50 = 830 nM T98397 C87XGZ 135964413 IC50 = 900 nM T98397 CV5TM7 135964419 IC50 = 23000 nM T98397 CM2W7G 135964420 IC50 = 2400 nM T98397 C3LWJ1 136002235 Ki = 7.01 nM T98397 C3Z2KF 136016315 IC50 = 68 nM T98397 CJ7ES6 136016316 IC50 = 6.3 nM T98397 C24FWM 136016317 IC50 = 5.5 nM T98397 C9SMI1 136016318 IC50 = 10 nM T98397 CMG1F8 136016319 IC50 = 4.7 nM T98397 C1GE3H 136016320 IC50 = 10 nM T98397 C2BV4Z 136016332 Ki = 750 nM T98397 CRE1J7 136023972 Ki = 2.5 nM T98397 CUM6S7 136030572 Ki = 660 nM T98397 CS8G9H 136035435 IC50 = 57.54 nM T98397 CT43BO 136035725 IC50 = 2000 nM T98397 CP7R4E 136035728 Ki = 50 nM T98397 COZ38B 136035729 Ki = 46 nM T98397 C20FIT 136035730 Ki = 150 nM T98397 CT3EH0 136035731 Ki = 24 nM T98397 C3PN0F 136035732 Ki = 26 nM T98397 C95NEC 136035733 Ki = 20 nM T98397 C9GWN1 136035734 Ki = 70 nM T98397 CV8L0C 136035735 Ki = 45 nM T98397 CTS1Q2 136035736 Ki = 260 nM T98397 CIJ7V5 136040460 IC50 = 575.44 nM T98397 C5KNS8 136041243 Ki = 5.5 nM T98397 CXFL78 136044124 IC50 = 7300 nM T98397 C2NU7R 136044125 Ki = 27 nM T98397 C4SD7H 136044126 Ki = 37 nM T98397 C1O9KB 136044135 IC50 = 2500 nM T98397 COQ8S5 136044136 IC50 = 2400 nM T98397 C2WX5Z 136044192 Ki = 150000 nM T98397 CT0NK9 136046104 IC50 > 40000 nM T98397 C9BEL8 136046118 IC50 = 128.82 nM T98397 CA1R9P 136046152 IC50 > 5000000 nM T98397 C6CMD5 136046154 IC50 = 100000 nM T98397 C3G9TR 136055872 Ki = 0.124 nM T98397 C8DBH4 136055873 Ki = 1.31 nM T98397 C9JB2N 136056457 IC50 = 90 nM T98397 C2A1FJ 136056459 IC50 = 2400 nM T98397 CK8U2L 136056477 IC50 > 200000 nM T98397 CB2Z1R 136056479 IC50 = 346.74 nM T98397 C3CZ2T 136056481 IC50 = 4265.8 nM T98397 CJGD84 136056484 IC50 = 2344.23 nM T98397 C1NF5D 136056496 IC50 = 39.81 nM T98397 C2C3KN 136056497 IC50 = 758.58 nM T98397 CVB02A 136056498 IC50 = 158.49 nM T98397 CI8Y2B 136056504 IC50 = 151.36 nM T98397 C37FHA 136056534 IC50 = 24547.09 nM T98397 CB49DE 136056552 IC50 = 776.25 nM T98397 CMIE21 136056553 IC50 = 616.6 nM T98397 CW5M6L 136056554 IC50 = 1778.28 nM T98397 CX3ZK5 136056555 IC50 = 537.03 nM T98397 C48NQT 136056556 IC50 = 218.78 nM T98397 CB4NK0 136056557 IC50 = 19952.62 nM T98397 C58WHM 136056558 IC50 = 1288.25 nM T98397 CG0Y2S 136056559 IC50 = 2884.03 nM T98397 C8Q3DW 136056560 IC50 = 12882.5 nM T98397 C1I0XW 136056561 IC50 = 169.82 nM T98397 CSXK85 136056562 IC50 = 478.63 nM T98397 C1MI7G 136056563 IC50 = 912.01 nM T98397 CH42AR 136056564 IC50 = 218.78 nM T98397 CLA9T6 136056565 IC50 = 16218.1 nM T98397 C04DLQ 136056566 IC50 = 501.19 nM T98397 C1TZ6C 136056567 IC50 = 25118.86 nM T98397 C2QY5N 136056568 IC50 = 478.63 nM T98397 CSN78B 136056569 IC50 = 645.65 nM T98397 CNV6C1 136056571 IC50 = 338.84 nM T98397 CZP8L0 136056572 IC50 = 36.31 nM T98397 C0UW9J 136056573 IC50 = 57.54 nM T98397 CY98WL 136056574 IC50 = 8.913 nM T98397 C3C2UZ 136056575 IC50 = 309.03 nM T98397 C8OE2B 136056577 IC50 = 42.66 nM T98397 CLA0D9 136056578 IC50 = 851.14 nM T98397 C6LN4D 136056579 IC50 = 676.08 nM T98397 CGUN14 136056580 IC50 = 169.82 nM T98397 CT4HN5 136056581 IC50 = 77.62 nM T98397 CT09OV 136056582 IC50 = 288.4 nM T98397 CFB50E 136056583 IC50 = 3548.13 nM T98397 CNHA09 136056585 IC50 = 977.24 nM T98397 CO63FU 136056586 IC50 = 11748.98 nM T98397 CBC54D 136056587 IC50 = 588.84 nM T98397 CFS09P 136056588 IC50 = 3801.89 nM T98397 CZ3RH1 136056589 IC50 = 74.13 nM T98397 CZ1X2A 136056590 IC50 = 5128.61 nM T98397 CBZ4O2 136056591 IC50 = 75.86 nM T98397 C53CBX 136056592 IC50 = 120.23 nM T98397 C3WY8H 136056593 IC50 = 67.61 nM T98397 CX21ZU 136056594 IC50 = 1737.8 nM T98397 CY78AO 136056595 IC50 = 190.55 nM T98397 C03MBN 136056596 IC50 = 933.25 nM T98397 CWJ59P 136056597 IC50 = 9332.54 nM T98397 CO0Z3R 136056598 IC50 = 316.23 nM T98397 CC1X6R 136056599 IC50 = 1348.96 nM T98397 C1J6RP 136056600 IC50 = 501.19 nM T98397 CLO9D8 136074285 IC50 = 42 nM T98397 CA0MF4 136074288 IC50 = 180000 nM T98397 CA43SM 136074303 Ki = 16700 nM T98397 CQ8NI7 136074304 Ki = 18 nM T98397 CPB97G 136074305 Ki = 79 nM T98397 C5J7FO 136074306 Ki = 57 nM T98397 C43BWK 136079589 Ki = 0.224 nM T98397 CNYR57 136079591 Ki = 0.072 nM T98397 CO6PC1 136079592 Ki = 0.041 nM T98397 CGN7B6 136079595 Ki = 0.042 nM T98397 CS67MO 136086679 IC50 = 436.52 nM T98397 C4IHJ5 136086682 IC50 = 1862.09 nM T98397 CRQ1C9 136086683 IC50 = 1659.59 nM T98397 C8UT1O 136086687 IC50 = 549.54 nM T98397 CV7EZ1 136086688 IC50 = 1202.26 nM T98397 C3V2SY 136086689 IC50 = 3388.44 nM T98397 C6ASQ1 136086690 IC50 = 3090.3 nM T98397 CTUD51 136086695 IC50 = 229.09 nM T98397 C07EVL 136086696 IC50 = 7079.46 nM T98397 C5WB6Y 136086697 IC50 = 229.09 nM T98397 CT5DV0 136086701 IC50 = 1071.52 nM T98397 CUK06X 136086702 IC50 = 190.55 nM T98397 CX24JH 136086703 IC50 = 416.87 nM T98397 CGH3O5 136086704 IC50 = 1737.8 nM T98397 C0A9OD 136086705 IC50 = 340 nM T98397 CQD8V9 136086706 IC50 = 933.25 nM T98397 CC98EH 136171347 IC50 = 770000 nM T98397 CVN97X 136171349 IC50 = 270 nM T98397 CAW95O 136209381 IC50 = 83000 nM T98397 CIKB26 136209383 IC50 = 31000 nM T98397 C5KAG4 136215366 Ki = 58 nM T98397 CX8OU5 136215367 Ki = 120000 nM T98397 C59LSN 136215368 Ki = 150000 nM T98397 CFU5N6 136227773 Ki = 3.3 nM T98397 CFUY16 137633842 IC50 = 1100 nM T98397 CS23KQ 137635618 IC50 = 120 nM T98397 CU8YX6 137643005 IC50 = 2300 nM T98397 CQUY83 137652218 IC50 = 480 nM T98397 C9JT1N 137655519 IC50 = 140 nM T98397 C2XOC5 139207781 IC50 = 3200 nM T98397 CWP60F 139207782 IC50 = 1700 nM T98397 CXA28V 139207783 IC50 = 800 nM T98397 C6YT3Z 139207784 IC50 = 1300 nM T98397 C6Q1IA 139207785 IC50 = 1800 nM T98397 C7F3BA 139207786 IC50 = 3500 nM T98397 CM5LU7 139207787 IC50 = 260 nM T98397 CP1Z3F 139207788 IC50 = 600 nM T98397 CA4TE7 139207789 IC50 = 460 nM T98397 CE3SK8 139207790 IC50 = 1000 nM T98397 C40VYJ 139207791 IC50 = 2200 nM T98397 C5FY6W 139207792 IC50 = 260 nM T98397 C08FCY 155512308 IC50 = 2800 nM T98397 CZ1V3R 155515740 IC50 = 3800 nM T98397 CEH1X0 155518060 IC50 = 1200 nM T98397 CM90WB 155518938 IC50 = 6000 nM T98397 CRJ78M 155526315 IC50 = 600 nM T98397 C8PVC4 155526575 IC50 = 700 nM T98397 CIR7C8 155526581 IC50 = 1580 nM T98397 CDUK46 155526588 IC50 = 390 nM T98397 C8EBQ2 155527133 IC50 = 1280 nM T98397 CITJ48 155527974 IC50 = 740 nM T98397 CTBW58 155529526 IC50 = 1970 nM T98397 CAL6V4 155534048 IC50 = 130 nM T98397 CK8TW2 155546343 IC50 = 2.4 nM T98397 CLKN30 155552168 IC50 = 450 nM T98397 C2PEB7 155552374 IC50 = 870 nM T98397 CX35ZM 155553154 IC50 = 470 nM T98397 CH61LS 155555206 IC50 = 130 nM T98397 C0HY3J 155555552 IC50 = 7300 nM T98397 CXWQ12 155560218 IC50 = 52000 nM T98397 CBT41K 155562260 IC50 = 98000 nM T98397 C89RGX 155562924 IC50 = 1300 nM T98397 C5SG2Z 155567595 IC50 = 560 nM T98397 CZ29BE 155568697 IC50 = 1650 nM T98397 CK58NL 135722143 IC50 = 120.23 nM T98397 CI2X8A 136056448 IC50 = 1445.44 nM T98397 C3PWK2 136056452 IC50 = 1148.15 nM T98397 D00IBG 643976 IC50 > 500000 nM T98397 D06DIH 158376 IC50 > 200000 nM T98397 D07LML 445504 Ki = 1100000 nM T98397 D07LSP 135438608 Ki = 7 nM T98397 D09QPT 135838247 Ki = 5400 nM T98397 D0CZ3C 65063 Ki = 3000 nM T98397 D0F1LA 446468 Ki = 49000 nM T98397 D0F2VL 135838221 Ki = 7000 nM T98397 D0G6CU 437081 Ki = 260 nM T98397 D0I0OH 8642 Ki = 14 nM T98397 D0Q0EB 135400203 IC50 = 39.81 nM T51076 D07TOK 46188928 IC50 = 24 nM T51076 D0AF6O 71731823 IC50 = 46 nM T51076 D01HKZ 57345941 IC50 < 3 nM T51076 D0E3TC 44259 IC50 = 0.22 nM T51076 D0FA6S 54576299 IC50 = 0.83 nM T51076 D0O0LS 25141092 IC50 < 10 nM T51076 CJ3Q5R 3666186 IC50 > 10000 nM T51076 CPZY43 5121984 IC50 > 50000 nM T51076 C7SCJ2 9206007 IC50 = 25960 nM T51076 CUJR40 10062694 EC50 = 30 nM T51076 C36EVF 11705812 IC50 = 29 nM T51076 C5VPH9 16129448 IC50 = 1600 nM T51076 C7HOI0 20907256 IC50 > 81010 nM T51076 CJPK63 20907257 IC50 > 3000 nM T51076 C7YG1N 24759534 IC50 = 380 nM T51076 CC69VF 24816435 IC50 = 40 nM T51076 CJ0CU5 24825841 IC50 = 4.35 nM T51076 C0KMW8 24937716 IC50 = 4 nM T51076 C5WG1H 24937847 IC50 = 3 nM T51076 C76PSW 44518384 IC50 = 11 nM T51076 C6LP9V 44518674 IC50 = 19 nM T51076 C36KYB 44520611 IC50 = 8 nM T51076 CZH80Q 44520612 IC50 = 980 nM T51076 CM39AU 46275360 IC50 = 20690 nM T51076 CLS29B 46872626 IC50 > 10000 nM T51076 C1EVX0 58063117 IC50 = 1300 nM T51076 CSG5T1 58335664 IC50 = 2 nM T51076 CXJ63M 59603829 IC50 = 120 nM T51076 CQEU96 59603842 IC50 = 13 nM T51076 CBZ9L7 66675408 IC50 > 10000 nM T51076 C37NKO 67129970 IC50 > 10000 nM T51076 CK80LJ 67130050 IC50 > 10000 nM T51076 CV63UL 67240318 IC50 > 10000 nM T51076 CK31BI 67330085 IC50 <= 5 nM T51076 C0VJW8 68545858 IC50 = 6 nM T51076 C7GRV2 68755406 IC50 > 10000 nM T51076 C5DGR9 69036886 IC50 = 157 nM T51076 CX7Z2M 70688180 IC50 = 97 nM T51076 CK2V4F 70690202 IC50 = 1900 nM T51076 C1V3NZ 73425588 IC50 = 4.38 nM T51076 CIQ5D8 74627727 IC50 = 142.1 nM T51076 C1HW4B 89735655 IC50 = 1400 nM T51076 CI4N8P 91801232 IC50 = 503 nM T51076 C3PAN1 117967296 IC50 = 25000 nM T51076 CK9ZY1 117967567 IC50 = 2300 nM T51076 C5M6NG 117968174 IC50 = 7100 nM T51076 CE86QC 118128728 IC50 = 2483.7 nM T51076 C0TMZ8 118167692 IC50 = 1.1 nM T51076 CLH8X7 118189551 IC50 = 2.3 nM T51076 CL0YO5 118443595 IC50 = 8.4 nM T51076 CU3K0B 118456253 IC50 = 4100 nM T51076 C60TWO 118665627 IC50 = 3.9 nM T51076 CDK5G4 118687517 IC50 = 5.9 nM T51076 CPK47S 118868365 IC50 = 2.2 nM T51076 CN4X0C 121231414 IC50 = 30.2 nM T51076 CO19NG 121272655 IC50 = 68160 nM T51076 CA6Z4R 121272745 IC50 > 81010 nM T51076 C08KEM 122179540 IC50 = 100 nM T51076 CQ43XF 122179541 IC50 = 230 nM T51076 C2TXZ9 122179542 IC50 = 75 nM T51076 CXS1Y6 122179543 IC50 = 40 nM T51076 CPF2L7 122179544 IC50 = 3 nM T51076 C3NJ6T 122179545 IC50 = 20 nM T51076 C3AJ4C 122179546 IC50 = 1 nM T51076 CG0RP7 122179547 IC50 < 1 nM T51076 C1A0SQ 122179548 IC50 = 2 nM T51076 CC83HO 123131777 IC50 > 81000 nM T51076 C1X6FJ 134693894 IC50 = 18 nM T51076 CY4D8I 135566504 Ki = 828.3 nM T51076 CG3UZ1 135927974 Ki > 1000 nM T51076 CXC69T 137321158 IC50 = 7 nM T51076 CWC49K 137321210 IC50 > 1000 nM T51076 CO2P6J 137632400 IC50 = 120000 nM T51076 CW6G0M 137633567 IC50 = 51000 nM T51076 C7P8DL 137633612 IC50 > 81010 nM T51076 CI1E8V 137634241 IC50 = 7700 nM T51076 C2YZA9 137634804 IC50 > 81010 nM T51076 CS1J9F 137638576 IC50 > 81010 nM T51076 C1BC7X 137638843 IC50 > 81010 nM T51076 C0NKR4 137640958 IC50 > 81010 nM T51076 CB3R4E 137641283 IC50 = 80270 nM T51076 CPK38A 137642417 IC50 > 81010 nM T51076 CW3K1R 137642682 IC50 = 38500 nM T51076 CO0A5Z 137643316 IC50 = 38550 nM T51076 CHQ75A 137644894 IC50 = 80020 nM T51076 C0IS6J 137647123 IC50 = 81160 nM T51076 C93MXU 137648253 IC50 = 47860 nM T51076 CE0LZ1 137648904 IC50 > 27000 nM T51076 C8F4ZH 137649400 IC50 > 81010 nM T51076 CQ98LD 137650528 IC50 > 81010 nM T51076 C9YQS6 137652057 IC50 > 81010 nM T51076 C29VEU 137652242 IC50 > 81010 nM T51076 CH9BQ6 137653271 IC50 > 81010 nM T51076 C48CER 137655170 IC50 > 81010 nM T51076 CD05EL 137655675 IC50 = 70240 nM T51076 CP87FM 137655709 IC50 > 81010 nM T51076 C2A1BD 137656463 IC50 > 81010 nM T51076 CYG87D 137656818 IC50 = 25140 nM T51076 CC4GR1 137657302 IC50 = 71720 nM T51076 CG5U3H 137657614 IC50 > 9001 nM T51076 CN3WV0 137657779 IC50 = 68750 nM T51076 C7E9YA 137658125 IC50 = 73070 nM T51076 CIJZ70 137658859 IC50 > 81010 nM T51076 C8GQ4F 137659402 IC50 = 58440 nM T51076 CYVK51 137659623 IC50 > 81010 nM T51076 CIC3L2 137659789 IC50 > 81010 nM T51076 CSWC68 137660376 IC50 > 9001 nM T51076 CJ0W9X 137660998 IC50 = 53490 nM T51076 CU9F5N 137661074 IC50 > 81010 nM T51076 CNRT47 139434032 EC50 = 1000 nM T51076 CIN6L7 139434035 EC50 = 330 nM T51076 CTFE03 139434036 EC50 = 180 nM T51076 CX9H4W 139434047 EC50 = 480 nM T51076 CU10QZ 139434077 EC50 = 510 nM T51076 CB6F5R 139434105 EC50 = 1400 nM T51076 C08MUD 139434127 EC50 = 190 nM T51076 C2MZ4L 139434198 EC50 = 220 nM T51076 C7W5MH 139434224 EC50 = 170 nM T51076 CXIT16 139434239 EC50 = 330 nM T51076 C2B8OV 139442846 EC50 = 90 nM T51076 CAJQ14 145964002 IC50 = 8.4 nM T51076 CVF4M6 145965985 IC50 = 1 nM T51076 C5MHK6 145967970 IC50 = 500 nM T51076 CK9C0H 145970062 IC50 = 5 nM T51076 CI85EU 145998085 IC50 = 790 nM T51076 CA10CQ 155512867 IC50 = 692.5 nM T51076 C2MD1Q 155513187 IC50 > 10000 nM T51076 C5B2AX 155513312 IC50 = 6.52 nM T51076 CZMD64 155514443 IC50 = 934.9 nM T51076 CB5T9G 155515436 IC50 = 215.4 nM T51076 CUHZ87 155516883 IC50 > 1000 nM T51076 CIU1T6 155518465 IC50 = 14.55 nM T51076 CO63MP 155519543 IC50 = 2.95 nM T51076 CBG4P0 155524103 IC50 = 8.84 nM T51076 CN6C2T 155528463 IC50 = 5.71 nM T51076 C0HW7F 155530527 IC50 > 1000 nM T51076 CP5IW9 155530600 IC50 > 1000 nM T51076 C3MC2P 155532434 IC50 = 66.98 nM T51076 CNE6A3 155532801 IC50 = 11.46 nM T51076 C2KAU0 155533663 IC50 = 16.8 nM T51076 C75AKY 155533695 IC50 < 10 nM T51076 C3PWI1 155534046 IC50 > 1000 nM T51076 CTXK93 155535665 IC50 = 158.9 nM T51076 C14SEB 155535950 IC50 = 46.3 nM T51076 CV9D5J 155536164 IC50 = 129 nM T51076 C3O6WX 155540330 IC50 > 1000 nM T51076 C76NKG 155543431 IC50 > 1000 nM T51076 CRV40J 155546026 IC50 = 44.58 nM T51076 C8AG4U 155550655 IC50 = 6.1 nM T51076 C2RQT8 155550913 IC50 < 10 nM T51076 C9MJL5 155551408 IC50 = 364.2 nM T51076 CYD1C7 155560599 IC50 > 1000 nM T51076 CBG9Z1 155562952 IC50 = 278 nM T51076 C0WZ9S 155563842 IC50 > 1000 nM T51076 CWR4O5 155565233 IC50 = 4.1 nM T51076 CRFW02 155566430 IC50 = 11.48 nM T51076 C0V7SM 155567015 IC50 > 1000 nM T51076 D0K5UF 72710568 IC50 = 18 nM T51076 D0N4LR 53469448 IC50 = 1115 nM T51076 D0O8AR 16097523 IC50 = 7.2 nM T51076 D0R2WK 16038120 EC50 > 1000 nM T54582 D00SQN 12136798 IC50 = 2100 nM T54582 D0H9SX 6914657 IC50 = 0.0301 nM T54582 D0Y1NC 148198 IC50 = 2 nM T54582 D0W9NH 2746 IC50 > 2000 nM T54582 C84NBV 215946 IC50 > 100000 nM T54582 C8US3L 293813 IC50 = 13000 nM T54582 C4WE3F 573291 IC50 = 38000 nM T54582 C92LZV 649594 IC50 = 91000 nM T54582 CUN5Q0 671605 IC50 = 13000 nM T54582 CJH2Q5 725650 IC50 = 1400 nM T54582 CVP4J2 790256 IC50 = 1000 nM T54582 CK90BW 804302 IC50 > 10000 nM T54582 CT70LU 887835 IC50 = 1600 nM T54582 CH35SZ 892011 IC50 = 630 nM T54582 CW8O9Z 1246974 IC50 = 860 nM T54582 CN75RQ 1250324 IC50 = 83000 nM T54582 C3J6TG 1251536 IC50 = 10300 nM T54582 CC4ON3 2229701 IC50 = 1900 nM T54582 C9N2PM 2537535 IC50 = 950 nM T54582 CO75GZ 2729251 IC50 < 5000 nM T54582 CNDI74 2803101 IC50 > 10000 nM T54582 CQ6TG1 2803102 IC50 = 7 nM T54582 CIHE54 2810548 IC50 = 150 nM T54582 C6Z4QL 2952642 IC50 = 1000 nM T54582 CBY8S1 2982781 IC50 > 100000 nM T54582 CSE8Y2 3491502 IC50 > 100000 nM T54582 C7U1ZB 4138811 IC50 = 5300 nM T54582 C64RVX 4456032 IC50 > 2000 nM T54582 C5H0IM 4786962 IC50 > 10000 nM T54582 C48JVZ 7208642 IC50 = 1000 nM T54582 C68QTV 9268468 IC50 = 26000 nM T54582 CG89YS 9938280 IC50 = 0.31 nM T54582 C5EXB3 13371091 IC50 = 170 nM T54582 CK5M7R 16774572 IC50 > 100000 nM T54582 CBG7S8 17018925 IC50 = 610 nM T54582 C6V1KQ 17464539 IC50 > 100000 nM T54582 C38QTW 18847535 IC50 = 1500 nM T54582 C5OPD6 20784945 IC50 = 90000 nM T54582 CCR1B3 20956142 IC50 = 8000 nM T54582 C0GR1O 22576752 IC50 = 242.7 nM T54582 C24PYD 25230395 IC50 = 38.5 nM T54582 CC8H7S 25519181 IC50 = 670 nM T54582 C9N1EM 26422900 IC50 = 420 nM T54582 C6H5ZS 26592135 IC50 = 36000 nM T54582 CN87FL 26775756 IC50 > 10000 nM T54582 CDXW40 31826481 IC50 = 940 nM T54582 CKI7C0 32220273 IC50 = 290 nM T54582 C9VI4K 32229604 IC50 = 3200 nM T54582 CG72AM 35523911 IC50 > 10000 nM T54582 CAK29J 37591481 IC50 = 780 nM T54582 C6H0IB 38754740 IC50 = 1500 nM T54582 CHD1V9 38754764 IC50 = 640 nM T54582 CND7Q9 40008574 IC50 = 220 nM T54582 C3CG1S 40075059 IC50 = 5000 nM T54582 CA34IQ 40108106 IC50 > 100000 nM T54582 CV8R7Z 44123681 IC50 = 0.2 nM T54582 CX40QY 44136054 IC50 = 2.4 nM T54582 CKLB25 44136825 IC50 = 0.3 nM T54582 CZ7TN3 44137619 IC50 = 1.1 nM T54582 C90XTB 44819697 IC50 = 3 nM T54582 CIYK50 45793870 IC50 = 50000 nM T54582 CSKR68 46077567 IC50 = 320 nM T54582 CE4UP5 46184343 IC50 = 49 nM T54582 CRFC05 46184581 IC50 = 8.2 nM T54582 C4LS1O 46628293 IC50 = 13000 nM T54582 C40PAI 47084288 IC50 = 41.8 nM T54582 C35DAM 47194703 IC50 = 850000 nM T54582 CHLT07 49836081 IC50 = 1.4 nM T54582 CDO5F0 49855415 IC50 = 250 nM T54582 C2BD7G 49855416 IC50 = 31 nM T54582 CD34NT 49855417 IC50 = 0.45 nM T54582 C6ODP0 49855418 IC50 = 12 nM T54582 C71KGT 49855419 IC50 = 1.2 nM T54582 CP1H0S 49855608 IC50 = 2.6 nM T54582 CR8S2L 49855609 IC50 = 13 nM T54582 CS53UR 49855610 IC50 = 56 nM T54582 C0T2ZW 49855611 IC50 = 12 nM T54582 CB4U8K 49855612 IC50 = 660 nM T54582 C0RZ4X 49855807 IC50 = 210 nM T54582 CK2J4R 49855808 IC50 = 2.9 nM T54582 CDA9V2 49855809 IC50 = 950 nM T54582 C5RP3W 49855810 IC50 = 2600 nM T54582 CC04ZN 49855811 IC50 > 10000 nM T54582 C3S7DO 49856003 IC50 > 10000 nM T54582 CKM4D5 49857135 IC50 = 0.79 nM T54582 CN06AI 49857137 IC50 = 12 nM T54582 C0J4LA 49857139 IC50 = 3.8 nM T54582 CC30NV 49857141 IC50 = 1200 nM T54582 CS7C2X 49857327 IC50 = 90 nM T54582 CL61NM 49857329 IC50 > 10000 nM T54582 C04QXN 49857330 IC50 = 600 nM T54582 C7DZ6G 49857532 IC50 > 10000 nM T54582 C9CVX1 49857533 IC50 = 330 nM T54582 C6C7IA 49857727 IC50 = 15 nM T54582 CAIY63 49857728 IC50 > 10000 nM T54582 CQ2TR4 49857729 IC50 = 420 nM T54582 C2D3GA 49857730 IC50 = 6.1 nM T54582 CDSJ17 49857731 IC50 = 4.2 nM T54582 CFH71A 49857732 IC50 = 1.3 nM T54582 CA0OP4 49857913 IC50 = 1.9 nM T54582 CGSW94 49857914 IC50 = 1.5 nM T54582 CK9G1D 49857915 IC50 = 110 nM T54582 C3LH9J 49857916 IC50 = 40 nM T54582 C9G0JI 49857917 IC50 = 0.55 nM T54582 CES3F4 49857918 IC50 = 11 nM T54582 CXP48R 49858108 IC50 = 25 nM T54582 CW15YT 49858109 IC50 = 3.6 nM T54582 C3VB8F 49858110 IC50 = 130 nM T54582 CT9N1R 49858111 IC50 > 10000 nM T54582 CW6NZ3 49858112 IC50 = 85 nM T54582 CVJ2X9 49858298 IC50 = 34 nM T54582 CFW3J4 49858299 IC50 = 49 nM T54582 C4EB3K 49858300 IC50 = 98 nM T54582 CW3SR2 49858301 IC50 = 150 nM T54582 CW9XG3 49858302 IC50 = 30 nM T54582 CE8NJ3 50913360 IC50 > 100000 nM T54582 C1K2VG 50913515 IC50 > 100000 nM T54582 CRF0C3 50914609 IC50 = 210 nM T54582 CY2M3C 50914751 IC50 = 14 nM T54582 C1PH3N 51031047 IC50 = 20300 nM T54582 CA86SC 51194992 IC50 = 1100 nM T54582 CQC9N3 51264526 IC50 = 25 nM T54582 CZ94FX 52358357 IC50 = 80 nM T54582 C0O3FD 53012900 IC50 = 3800 nM T54582 C3DP4L 56680013 IC50 = 0.3 nM T54582 CS8R7Y 56837162 IC50 = 21 nM T54582 CYU69S 56924625 IC50 = 2.4 nM T54582 CR1L6W 56928256 IC50 = 7.5 nM T54582 C6P1LZ 56928663 IC50 = 30 nM T54582 CU6N7O 56928682 IC50 = 2.5 nM T54582 C8G7MV 56928784 IC50 = 2 nM T54582 C63AVQ 56929155 IC50 = 49 nM T54582 C6LA8E 56929163 IC50 = 2.6 nM T54582 CGXK64 56929167 IC50 = 4.4 nM T54582 C0FRB5 56929168 IC50 = 3.6 nM T54582 C54GXP 56929243 IC50 = 60 nM T54582 CEP57G 56929356 IC50 = 1.7 nM T54582 C8RK6Q 56929542 IC50 = 0.6 nM T54582 CUW67B 56929624 IC50 = 1.2 nM T54582 CHLE49 56929641 IC50 = 1.9 nM T54582 CNJ71C 56943182 IC50 = 1300 nM T54582 CPAU51 56943206 IC50 = 14 nM T54582 CT0V7Y 56943314 IC50 = 1500 nM T54582 CCF81W 56943316 IC50 > 10000 nM T54582 CT8I2N 56943317 IC50 = 37 nM T54582 CPFK26 56943401 IC50 = 4.5 nM T54582 C25ODG 57509628 Ki = 9 nM T54582 CKN73A 57509646 Ki = 7.9 nM T54582 C1FRH4 57509651 Ki = 4.7 nM T54582 CXZ1I4 57509662 Ki = 11 nM T54582 C7JZF8 57509669 Ki = 13 nM T54582 CH7Y5L 57509676 Ki = 14 nM T54582 CM5CE4 57509679 Ki = 14 nM T54582 CHIS60 57509685 Ki = 16 nM T54582 C58AYK 57509693 Ki = 17 nM T54582 CO34BS 57509699 Ki = 19 nM T54582 CLE32W 57509712 Ki = 23 nM T54582 C6XK1I 57509717 Ki = 24 nM T54582 CGLX74 57509834 Ki = 104 nM T54582 C43CEU 57509874 Ki = 560 nM T54582 C6GPH9 57509876 Ki = 19 nM T54582 C45HQP 57509914 Ki = 7.5 nM T54582 CKH61U 57509918 Ki = 58 nM T54582 CE80WD 57509943 Ki = 23 nM T54582 CNOT61 57509956 Ki = 3 nM T54582 CI9G8Y 57509958 Ki = 19 nM T54582 CA0RQ6 57509971 Ki = 1.6 nM T54582 C8CZ6I 57509986 Ki = 5.4 nM T54582 CWA5E1 57510022 Ki = 15 nM T54582 C6BH9L 57510023 Ki = 1 nM T54582 CHP41X 57510036 Ki = 13 nM T54582 CZS0K6 57510184 Ki = 57 nM T54582 CP6V7X 57510215 Ki = 4.9 nM T54582 CMY38S 57510390 Ki = 350 nM T54582 C5QN4J 57510612 Ki = 18 nM T54582 C73HKY 57527898 Ki = 2200 nM T54582 CWT6O0 57723146 IC50 > 100000 nM T54582 CZV9X5 59053520 IC50 = 19 nM T54582 C4LPO6 59053774 IC50 = 80000 nM T54582 C5EMD0 66608900 IC50 = 100 nM T54582 COV13X 66609141 IC50 > 10000 nM T54582 CU3SR0 66609318 IC50 = 1900 nM T54582 CH84WB 66609481 IC50 = 1 nM T54582 C1JV7U 66609540 IC50 = 6 nM T54582 C8X0CH 66609607 IC50 = 10 nM T54582 CSWU38 66609622 IC50 = 20 nM T54582 C5GK6W 66609666 IC50 = 60 nM T54582 CX3L8W 66609690 IC50 = 4800 nM T54582 C6HVF3 66609743 IC50 = 610 nM T54582 C7IMG8 66609911 IC50 = 19 nM T54582 COQ01G 66610004 IC50 = 54 nM T54582 CPZ2E3 66610017 IC50 = 26 nM T54582 COQ4E0 66610019 IC50 = 9 nM T54582 CR4TD9 66610060 IC50 = 1900 nM T54582 CJQ1K5 66610067 IC50 = 3 nM T54582 C6GIU4 66610210 IC50 = 59 nM T54582 CRG3E9 66610246 IC50 = 28 nM T54582 C9BY3S 66610338 IC50 = 4 nM T54582 C0YM2A 66610342 IC50 = 8 nM T54582 C1W6FK 66610365 IC50 = 4 nM T54582 CB12AN 66610375 IC50 = 24 nM T54582 CP93XE 66610384 IC50 > 2000 nM T54582 C0XB3J 66610415 IC50 = 11 nM T54582 CMQF12 66610527 IC50 = 7 nM T54582 C5VDX7 66610553 IC50 > 10000 nM T54582 CSP21O 66610560 IC50 = 7 nM T54582 C0V9KB 66610600 IC50 > 10000 nM T54582 C3N1PO 66610605 IC50 = 18 nM T54582 C29UKS 66610695 IC50 > 10000 nM T54582 CDPO14 66610702 IC50 = 9 nM T54582 CJ40XE 66610717 IC50 = 5 nM T54582 CEQA95 66610798 IC50 = 7 nM T54582 CJ7F8O 66610805 IC50 = 2000 nM T54582 CSV5K2 66610852 IC50 = 5 nM T54582 C1ZMK2 66610923 IC50 = 24 nM T54582 CS72TK 66610926 IC50 = 3 nM T54582 CA5ZW2 66610937 IC50 = 9 nM T54582 CC1FI7 66610941 IC50 = 17 nM T54582 C0AHJ2 66610946 IC50 = 12 nM T54582 CC4J9G 66611001 IC50 = 30 nM T54582 CA2H3P 66611008 IC50 = 10 nM T54582 C47TJK 66611017 IC50 = 14 nM T54582 C7M6XG 66611076 IC50 = 3 nM T54582 C7OD1P 66611088 IC50 = 470 nM T54582 C5R0KS 66611089 IC50 = 10 nM T54582 CVB4T1 66611375 IC50 = 7 nM T54582 CQ6K4U 66611591 IC50 > 10000 nM T54582 C72LEC 66613538 IC50 = 17 nM T54582 CJYZ32 66613587 IC50 = 12 nM T54582 C0CSL5 66613641 IC50 = 390 nM T54582 CFI5T8 66613669 EC50 = 1.2 nM T54582 C6JSA0 66613704 IC50 = 8 nM T54582 C52UTX 66613705 IC50 = 1000 nM T54582 C3QZ5E 66613756 IC50 = 7100 nM T54582 C42NIF 66613812 IC50 = 130 nM T54582 CF9OZ0 66613826 IC50 = 400 nM T54582 C40FBR 66613914 IC50 = 310 nM T54582 C7G2JC 66614012 IC50 = 150 nM T54582 C5TU3K 66614212 IC50 = 41 nM T54582 C3VXP7 66614375 IC50 = 28 nM T54582 CX26SR 66614451 IC50 > 2000 nM T54582 CGX2O7 66634544 IC50 > 2000 nM T54582 CTO6Z3 66870846 IC50 = 3300 nM T54582 CCX1F0 66871849 IC50 = 25000 nM T54582 CE1XW5 68090877 IC50 = 11 nM T54582 CUO2I1 68091015 IC50 = 1700 nM T54582 C7TR4I 68276577 IC50 = 10 nM T54582 CO0VH6 68276608 IC50 = 140 nM T54582 CJ6T0I 68276611 IC50 = 310 nM T54582 CW1C0I 68276677 IC50 = 7.7 nM T54582 CW2YH9 68276701 IC50 = 970 nM T54582 CT72LE 68276725 IC50 = 3 nM T54582 C62NZO 68276762 IC50 > 10000 nM T54582 CC1R6Y 68276866 IC50 = 370 nM T54582 CD68FL 68277248 IC50 = 8 nM T54582 C3RI1U 68277270 IC50 = 8 nM T54582 CHE9I2 68277271 IC50 = 8.2 nM T54582 C0I8FN 68277336 IC50 = 210 nM T54582 C9X3TF 68277348 IC50 = 43 nM T54582 C5F3YP 68277361 IC50 = 1900 nM T54582 CLI92H 68277393 IC50 = 8 nM T54582 CS6ZE2 68277395 IC50 = 41 nM T54582 CK74NM 68277440 IC50 = 12 nM T54582 CWJ9B3 68277492 IC50 = 7 nM T54582 CB3JP8 68277518 IC50 = 2 nM T54582 C3GM6V 68277541 IC50 = 3 nM T54582 C3D8WU 68277544 IC50 = 10 nM T54582 CK5V3O 68277611 EC50 = 1.1 nM T54582 CFZ2U7 68277645 IC50 = 5 nM T54582 CJ3N5T 68277668 IC50 = 16 nM T54582 CBV34D 68277935 IC50 = 9 nM T54582 CIYL98 68748359 Ki = 112 nM T54582 C9FVY5 70501112 IC50 > 100000 nM T54582 C51ZEX 70846229 IC50 = 34000 nM T54582 CRTC91 70983109 IC50 = 6.3 nM T54582 C5ZH7U 70984701 IC50 = 5.4 nM T54582 C7KJN8 71654714 IC50 = 13 nM T54582 CYD9P8 71654715 IC50 = 12 nM T54582 CWZ83T 71654716 IC50 = 1300 nM T54582 CB7H3S 71654717 IC50 = 600 nM T54582 CRM61V 71654718 IC50 = 14 nM T54582 C3W2YJ 71654788 IC50 = 52 nM T54582 CU50AM 71654790 IC50 = 33 nM T54582 CSV81U 71654791 IC50 = 47 nM T54582 CT34VN 71654792 IC50 = 103 nM T54582 C4BMW8 71654793 IC50 = 27 nM T54582 CCH0T6 71654852 IC50 = 6 nM T54582 CVEW58 71654853 IC50 = 5 nM T54582 C8WT4B 71654854 IC50 = 45 nM T54582 C6QT9L 71654855 IC50 = 100 nM T54582 C4CB5Y 71654856 IC50 = 11 nM T54582 CG1W6H 71654857 IC50 = 3 nM T54582 C43EHA 71654926 IC50 = 8 nM T54582 C6I3VF 71654927 IC50 = 142 nM T54582 CO6K8D 71654928 IC50 = 4 nM T54582 C8UVZ0 71654929 IC50 = 8 nM T54582 CJYU32 71654930 IC50 = 4 nM T54582 C1FNK2 71655701 IC50 = 146 nM T54582 CIA03F 71655702 IC50 > 2000 nM T54582 CF68KU 71655703 IC50 = 59 nM T54582 CQ1NY6 71655704 IC50 = 1400 nM T54582 CFU86J 71655705 IC50 = 7 nM T54582 CDO29V 71655706 IC50 = 40 nM T54582 CG4HW8 71655768 IC50 = 12 nM T54582 CL56VA 71655769 IC50 = 1500 nM T54582 CS2EN8 71655770 IC50 = 930 nM T54582 C6VRC0 71655771 IC50 = 1600 nM T54582 C7UA4I 71655772 IC50 = 680 nM T54582 CPB6T3 71655773 IC50 = 13 nM T54582 CMAW93 71711804 IC50 = 0.4 nM T54582 CO6Q3R 71715127 IC50 = 1.6 nM T54582 C6JS5H 71715183 IC50 = 9 nM T54582 CYR2J8 71715184 IC50 = 24 nM T54582 C6JS5R 71715185 IC50 = 10 nM T54582 CHS3X9 71715186 IC50 = 18 nM T54582 CIX79H 71715241 IC50 = 74 nM T54582 CQEH46 71720911 IC50 = 4 nM T54582 C4O6MY 71726495 IC50 = 150 nM T54582 C4Z7LR 71727359 IC50 = 7.1 nM T54582 C7TJI1 71727460 IC50 = 11 nM T54582 CB53IQ 71727461 IC50 = 11 nM T54582 CMF7Y2 71727572 IC50 = 78 nM T54582 CJ08QE 71727679 IC50 = 99 nM T54582 C0F4VI 71727680 IC50 = 190 nM T54582 C2SQ6K 71727682 IC50 = 2 nM T54582 C6S0WT 71727683 IC50 = 14 nM T54582 CLE15B 71727801 IC50 = 10 nM T54582 CV6QC1 71727805 IC50 = 58 nM T54582 C7WF2S 71727928 IC50 = 39 nM T54582 CE8R1D 71727929 IC50 = 98 nM T54582 C6USH8 71727930 IC50 = 20 nM T54582 C1W4DX 71727932 IC50 = 17 nM T54582 C36DNH 71727934 IC50 = 75 nM T54582 CJZR51 71728054 IC50 = 6 nM T54582 CBQJ18 71728058 IC50 = 170 nM T54582 C42HVX 71728060 IC50 = 15 nM T54582 CK9M4L 71728063 IC50 = 17 nM T54582 CJ5MF9 71728064 IC50 = 8 nM T54582 CHU65X 71734760 IC50 = 16 nM T54582 C3PGK9 71734761 IC50 = 12 nM T54582 CH70QW 71734762 IC50 = 1800 nM T54582 CT0BX5 71734763 IC50 = 28 nM T54582 CJ51WU 71734843 IC50 = 1800 nM T54582 CPH62M 71734921 IC50 = 11 nM T54582 C9O3BM 71817346 IC50 > 2000 nM T54582 C4KBF0 71817347 IC50 = 26 nM T54582 CO2SL0 71817348 IC50 = 44 nM T54582 CX53VW 71817349 IC50 = 83 nM T54582 C7MV4A 71817350 IC50 = 27 nM T54582 CC4SU1 71817351 IC50 = 31 nM T54582 CY04LE 71817500 IC50 = 10 nM T54582 C1OH2T 71817501 IC50 = 48 nM T54582 CJL7U9 71817502 IC50 = 58 nM T54582 C9DT3Z 71817503 IC50 = 71 nM T54582 CV9KO4 71817504 IC50 = 44 nM T54582 CC1OF5 71817505 IC50 = 28 nM T54582 CTM05H 71817663 IC50 = 770 nM T54582 CCA62S 71817664 IC50 = 38 nM T54582 CKB79E 71817665 IC50 = 59 nM T54582 CK6QM0 71817666 IC50 = 22 nM T54582 CG98JC 71817667 IC50 = 20 nM T54582 C86MPX 71817668 IC50 = 7.4 nM T54582 COF4Q6 71818013 IC50 = 410 nM T54582 CMU03Y 71818155 IC50 = 40 nM T54582 C4NEF1 71818156 IC50 = 150 nM T54582 CR4F3H 71818301 IC50 = 400 nM T54582 C3LNX4 71818452 IC50 = 1700 nM T54582 CTI9J5 71818453 IC50 = 1800 nM T54582 C5L0BE 71818454 IC50 = 3 nM T54582 C9CK8N 71818455 IC50 = 2 nM T54582 C2R4MQ 71818728 IC50 = 24 nM T54582 CN53KF 71818875 IC50 = 5 nM T54582 CX1JE4 71818876 IC50 = 3 nM T54582 C81YJE 71819015 IC50 = 3 nM T54582 CLA19N 71819152 IC50 = 1 nM T54582 C0QG8K 71819528 IC50 = 12 nM T54582 CUTA06 72163497 IC50 = 0.174 nM T54582 C03HSC 72545610 IC50 = 0.461 nM T54582 CH3QZ2 72546332 IC50 = 0.632 nM T54582 CC0P8V 72734880 IC50 = 4.4 nM T54582 C2PH4Y 72735060 IC50 = 3.2 nM T54582 CS3CX7 72735243 IC50 = 2.4 nM T54582 CT4QZ3 72771099 IC50 = 15 nM T54582 CAS03K 72945734 IC50 = 2.2 nM T54582 C5Y6LQ 72945736 IC50 = 5.4 nM T54582 CM3S9W 73346084 IC50 = 0.23 nM T54582 CSEF31 73350708 IC50 = 3 nM T54582 CGF24A 73355241 IC50 = 19 nM T54582 CCFI76 73890932 IC50 = 10 nM T54582 C9E0PX 76071764 IC50 = 5 nM T54582 C1Y7HC 76072411 IC50 = 5.1 nM T54582 C9G5QJ 76309996 IC50 = 3.6 nM T54582 C13TFQ 76310719 IC50 = 14000 nM T54582 CY0HD7 76311092 IC50 = 4.4 nM T54582 CZ2CL1 76311093 IC50 = 11 nM T54582 CVM9R7 76311094 IC50 = 750 nM T54582 C7JE1C 76311095 IC50 = 28 nM T54582 CAT65E 76311096 IC50 = 7.8 nM T54582 C3YV2L 76311097 IC50 = 1300 nM T54582 CKFT56 76313714 IC50 = 49.6 nM T54582 CQ6B2H 76314025 IC50 > 100000 nM T54582 C7AWE6 76314026 IC50 > 100000 nM T54582 CUS45M 76314338 IC50 = 3700 nM T54582 C7FXT3 76314339 IC50 = 6100 nM T54582 CGS0P6 76314340 IC50 > 100000 nM T54582 CX3LZ0 76314702 IC50 = 9.5 nM T54582 C0T5EU 76314704 IC50 > 2000 nM T54582 C0WZ2O 76317568 IC50 > 100000 nM T54582 CC4T2I 76317569 IC50 > 100000 nM T54582 C7Q6LG 76317926 IC50 = 5000 nM T54582 CVNI39 76317927 IC50 = 62000 nM T54582 CQP6N2 76317928 IC50 = 3400 nM T54582 CD85CI 76318275 IC50 = 10 nM T54582 CQ9K4T 76318276 IC50 = 1500 nM T54582 C67LZX 76320949 IC50 = 2.4 nM T54582 CPX27Y 76321629 IC50 > 100000 nM T54582 CD3T6K 76321630 IC50 = 4100 nM T54582 CDC2R5 76321977 IC50 > 2000 nM T54582 C1WR0Y 76321978 IC50 = 12 nM T54582 C7Y5QF 76321979 IC50 = 7.2 nM T54582 C2M8XT 76324594 IC50 = 133.2 nM T54582 CGA18X 76324595 IC50 = 11.8 nM T54582 CR15KG 76325247 IC50 = 21000 nM T54582 C1HJQ9 76325597 IC50 = 6.6 nM T54582 C7YKM5 76325598 IC50 > 2000 nM T54582 CO0GT1 76328151 IC50 = 22.8 nM T54582 C4BRX7 76328472 IC50 > 100000 nM T54582 CME4G5 76328800 IC50 > 100000 nM T54582 CA54CD 76328801 IC50 = 40000 nM T54582 C4KHG5 76328802 IC50 = 3100 nM T54582 CVQ72D 76328803 IC50 = 9100 nM T54582 CI1JV3 76328804 IC50 = 21000 nM T54582 CHBT56 76329161 IC50 = 3.8 nM T54582 CYTI04 76329162 IC50 = 7.6 nM T54582 CXY2H0 76329163 IC50 = 2 nM T54582 CZ9Q2S 76329164 IC50 = 49 nM T54582 CLW64K 76331860 IC50 = 4.4 nM T54582 CX3ON1 76332158 IC50 > 100000 nM T54582 CX8Q3T 76332475 IC50 = 1400 nM T54582 C34QRZ 76332476 IC50 > 100000 nM T54582 C04HRJ 76332822 IC50 > 2000 nM T54582 C9SX6E 76332823 IC50 = 4.7 nM T54582 C7MJA6 76332824 IC50 = 10 nM T54582 C3AJ2R 76332825 IC50 = 21 nM T54582 CZ2CQ7 76332826 IC50 = 8.8 nM T54582 C5T0RG 76335779 IC50 > 100000 nM T54582 C5SKO0 76336444 IC50 = 12 nM T54582 CR25FW 76336445 IC50 = 9 nM T54582 CGJM01 76336447 IC50 = 36 nM T54582 CNW57A 76336448 IC50 > 2000 nM T54582 CU5ZY3 86298751 IC50 = 4.9 nM T54582 CC8T1V 86305870 IC50 = 6.7 nM T54582 CWZ07E 86306023 IC50 = 7.8 nM T54582 C8RPT6 86920711 IC50 > 10000 nM T54582 C4ZR3M 89785082 IC50 = 47 nM T54582 C1QDJ0 89793388 IC50 = 4.3 nM T54582 CT9QL8 89793441 IC50 > 2000 nM T54582 CUS70D 89793496 IC50 = 10 nM T54582 CP7MZ2 89793516 IC50 = 39 nM T54582 C9X5OT 89793519 IC50 = 8 nM T54582 C0NS7R 89793535 IC50 = 7 nM T54582 C9OW4E 89795476 IC50 = 32 nM T54582 COZ7E3 89795479 IC50 = 21 nM T54582 C96EWN 89795484 IC50 = 19 nM T54582 CWO58S 89795501 IC50 = 11 nM T54582 CV7RP2 89795538 IC50 = 410 nM T54582 CC84ML 89795547 IC50 = 440 nM T54582 CIQ53M 89795553 IC50 = 8 nM T54582 CIR65O 89795596 IC50 = 88 nM T54582 C9SD1V 89795599 IC50 = 26 nM T54582 C6IG2Z 89795666 IC50 = 71 nM T54582 C6QAL3 89795694 IC50 = 110 nM T54582 C8C7IH 89795715 IC50 = 19 nM T54582 C5GQL0 89795796 IC50 = 43 nM T54582 C14ZXL 90011880 IC50 > 2000 nM T54582 CJ65EF 90012001 IC50 = 1.5 nM T54582 C9YC5X 90012681 IC50 = 19 nM T54582 C6KYB4 90012693 IC50 = 38.7 nM T54582 CI09NS 90012714 IC50 = 88 nM T54582 C36WKJ 90012746 IC50 = 300 nM T54582 C81JHW 90012820 IC50 = 410 nM T54582 C4F9YI 90012973 IC50 = 370 nM T54582 CG78UF 90013202 IC50 = 6.2 nM T54582 CIOZ97 90013255 IC50 = 20.4 nM T54582 CWY1R0 90655892 IC50 = 0.412 nM T54582 CMNF17 90655898 IC50 = 7.9 nM T54582 C6X5AH 90655899 IC50 = 10 nM T54582 CC1YK3 90655900 IC50 = 11 nM T54582 CP6MS3 118160922 IC50 = 84 nM T54582 CR3T9O 118193528 IC50 = 15 nM T54582 C89NET 118193544 IC50 = 34 nM T54582 CFH39Z 118621271 IC50 = 1.6 nM T54582 C18SWX 118621276 IC50 = 1 nM T54582 CR6AF2 118621278 IC50 = 41.2 nM T54582 C9A5WK 118621285 IC50 = 1.6 nM T54582 C9GCH6 118621295 IC50 = 4.4 nM T54582 CZR26D 118621302 IC50 = 4.8 nM T54582 CP07JL 118621306 IC50 = 5.3 nM T54582 C0WV1H 118621308 IC50 = 26.5 nM T54582 CF2Q7C 118621309 IC50 = 5.8 nM T54582 C9SY5J 118621333 IC50 = 31.2 nM T54582 CXU42D 118621370 IC50 = 3.5 nM T54582 C4VNM0 118621378 IC50 = 2.2 nM T54582 CXL76C 118621380 IC50 = 1.6 nM T54582 C4CSN8 118621388 IC50 = 47.8 nM T54582 CSU41F 118621392 IC50 = 6.5 nM T54582 CT0W3L 118621401 IC50 = 3.8 nM T54582 CHFL73 118621409 IC50 = 20.7 nM T54582 CYX1L5 118621411 IC50 = 6.9 nM T54582 CK87IQ 118621413 IC50 = 13.3 nM T54582 CHZ4T8 118726259 IC50 = 49 nM T54582 CPI1T8 118726260 IC50 = 5 nM T54582 CM8NK7 121499158 IC50 = 13 nM T54582 CDA13G 127027287 IC50 = 0.0509 nM T54582 C38BLA 127036410 IC50 = 1.1 nM T54582 CCTN19 127036434 IC50 = 7.6 nM T54582 CG1X0H 127036600 IC50 > 10000 nM T54582 C40MDL 127036749 IC50 > 10000 nM T54582 CGF5C1 131955128 IC50 = 10000 nM T54582 C9QYP1 132585220 Ki = 5.6 nM T54582 C8EAW2 132942960 IC50 = 66.9 nM T54582 C6DP2E 134130638 IC50 = 402 nM T54582 CS0N2O 134131947 IC50 = 16 nM T54582 CUIF45 134132017 IC50 = 14 nM T54582 CB51NS 134133237 IC50 = 6 nM T54582 C5IXF3 134136542 IC50 > 2000 nM T54582 CC57VG 134138726 IC50 > 2000 nM T54582 C21OUY 134139520 IC50 = 34 nM T54582 C9DBR7 134144418 IC50 > 1700 nM T54582 C14IWG 134146417 IC50 = 830 nM T54582 C7DX5U 134148567 IC50 = 423 nM T54582 CMTV01 134151719 IC50 > 2000 nM T54582 C6TML2 134152085 IC50 = 75 nM T54582 CFX51B 134154660 IC50 = 555.4 nM T54582 CQT9F3 134155188 IC50 > 2000 nM T54582 CXT0A2 134155658 IC50 = 473 nM T54582 C9UWD3 134155777 IC50 = 59 nM T54582 CU23AG 134562941 IC50 = 25.3 nM T54582 CP70KD 134814219 IC50 = 3.1 nM T54582 C9HKY8 134814226 IC50 < 1 nM T54582 C5IOY0 135567364 IC50 = 360000 nM T54582 C1F6MN 135998697 IC50 = 2800 nM T54582 CKS1C8 135998703 IC50 = 29 nM T54582 CL46PI 135998704 IC50 = 7200 nM T54582 C8NZP9 136224234 IC50 = 63 nM T54582 CHK6B8 136241658 IC50 = 62 nM T54582 CHYF09 137631675 IC50 = 230 nM T54582 CW3PD2 137632740 IC50 > 2000 nM T54582 C73PDL 137634086 IC50 = 31 nM T54582 CXV7Y4 137634585 Ki > 9000 nM T54582 C2ZLH6 137634772 IC50 > 2000 nM T54582 CX2A6H 137634973 Ki = 1.5 nM T54582 CPL42O 137635914 IC50 > 2000 nM T54582 CQ4FP7 137636752 IC50 = 18 nM T54582 C7OT8F 137637596 IC50 > 2000 nM T54582 C42PIU 137638406 IC50 > 2000 nM T54582 C5FGB4 137638429 IC50 > 2000 nM T54582 CP6NM0 137638747 IC50 > 2000 nM T54582 CF7XJ2 137640263 IC50 > 2000 nM T54582 CBQ7Z9 137640884 IC50 > 2000 nM T54582 COAB04 137641633 Ki = 2.5 nM T54582 CTJA80 137642143 IC50 > 2000 nM T54582 CA60BJ 137643597 Ki = 5.1 nM T54582 CEM38G 137644704 Ki > 8900 nM T54582 C1TKW9 137644960 IC50 > 2000 nM T54582 C84JEV 137645469 IC50 > 2000 nM T54582 CYA81D 137645509 IC50 > 2000 nM T54582 C6FPB8 137646630 IC50 > 2000 nM T54582 C4K5JC 137646664 IC50 > 2000 nM T54582 C3AIC9 137646743 IC50 > 2000 nM T54582 C6K2LI 137647251 Ki = 1.7 nM T54582 CI05DA 137648221 IC50 > 2000 nM T54582 CYEJ51 137649739 Ki = 21 nM T54582 CE70UO 137649967 Ki = 3.9 nM T54582 C9W6SR 137652347 Ki = 9.4 nM T54582 C7SUM3 137653261 IC50 = 550 nM T54582 C82RZU 137653956 IC50 = 116 nM T54582 C4C0YK 137654373 Ki = 1.9 nM T54582 CTN10F 137654680 IC50 > 2000 nM T54582 C79HAZ 137655524 IC50 > 2000 nM T54582 C2RKM4 137656021 IC50 = 190 nM T54582 C9PUK8 137656850 IC50 > 2000 nM T54582 C76UNZ 137656995 Ki = 4.3 nM T54582 CO5E2F 137658815 IC50 > 2000 nM T54582 C78QUS 137658818 Ki = 160 nM T54582 CE49SB 137659150 IC50 > 2000 nM T54582 C1C8HZ 137659782 IC50 > 2000 nM T54582 C6POG5 137660155 IC50 > 2000 nM T54582 CAOG59 137660901 IC50 > 2000 nM T54582 C2D6AS 145100135 IC50 = 702 nM T54582 CWBH61 145100138 IC50 = 544 nM T54582 CO91CW 145100139 IC50 = 1000 nM T54582 CP9UN1 145100143 IC50 = 52.7 nM T54582 CMV25K 145100151 IC50 = 120 nM T54582 CDGA06 145100154 IC50 = 149 nM T54582 CGS8V4 145100159 IC50 = 213 nM T54582 CKS8G5 145100160 IC50 = 285 nM T54582 CSCY68 145100164 IC50 = 181 nM T54582 CYAL61 145100169 IC50 = 873 nM T54582 C9X6YG 145704651 IC50 = 2.7 nM T54582 C4W0YE 145950607 IC50 = 470 nM T54582 C9SMA8 145950715 IC50 = 7 nM T54582 CRKM19 145950884 IC50 = 15 nM T54582 C5FU6W 145955202 IC50 = 220 nM T54582 C23ZAQ 145955356 IC50 = 18 nM T54582 C7B2EU 145956761 IC50 = 14 nM T54582 C3XI4V 145956897 IC50 = 14 nM T54582 C18ZGV 145959245 IC50 = 20 nM T54582 C1X5EO 145962694 IC50 = 19 nM T54582 CRU59M 145965285 IC50 = 10 nM T54582 CA1UB2 145965564 IC50 = 4.3 nM T54582 CTC68H 145971821 IC50 = 25 nM T54582 CYB37F 145971853 IC50 > 2500 nM T54582 C5BV9U 145973321 IC50 = 80 nM T54582 CHF69M 145974875 IC50 > 1000000 nM T54582 CZV97P 155512117 IC50 = 82.5 nM T54582 CT4VS3 155512474 IC50 > 100000 nM T54582 CF9N8E 155514200 IC50 = 362 nM T54582 C21JZQ 155514830 Ki = 0.2 nM T54582 C10CRP 155516301 IC50 = 99.6 nM T54582 CVY96R 155518484 Ki = 1.3 nM T54582 C8TX5M 155521513 Ki = 7.9 nM T54582 C8EB7S 155521647 IC50 = 14.42 nM T54582 CQLY73 155522530 IC50 = 16.41 nM T54582 CX57IN 155522805 IC50 = 9.78 nM T54582 CE8KO9 155524021 IC50 = 234.5 nM T54582 CK6NH5 155524184 IC50 = 9.7 nM T54582 CWC58R 155524192 IC50 = 31.54 nM T54582 C10QGH 155526016 IC50 = 780 nM T54582 CIJ9T2 155527509 IC50 = 12.28 nM T54582 CTU1Y5 155529354 Ki = 5.9 nM T54582 CMV42P 155532060 IC50 = 381 nM T54582 C3WJM2 155532586 IC50 = 54.8 nM T54582 CPCM60 155534374 IC50 = 24.53 nM T54582 C79CIB 155534963 Ki = 1.1 nM T54582 C0BH6F 155537916 IC50 = 5.08 nM T54582 CQ9N8E 155539825 IC50 = 16.54 nM T54582 CTAL05 155540057 IC50 = 28.39 nM T54582 C21OGH 155541419 IC50 = 715 nM T54582 C9GED2 155541536 IC50 = 31.32 nM T54582 C4T9YC 155542195 IC50 = 2500 nM T54582 CGP43Z 155543775 IC50 = 13.09 nM T54582 CF6LD7 155544739 IC50 = 5920 nM T54582 C1GXZ8 155545503 IC50 = 10.75 nM T54582 CE1D7Q 155546207 IC50 = 3900 nM T54582 CLT10R 155549611 IC50 = 10.53 nM T54582 CX8A0I 155553082 IC50 = 195 nM T54582 C1VLT7 155558605 IC50 = 9.47 nM T54582 C6Y1NX 155559135 IC50 = 17.77 nM T54582 CFS64P 155563379 Ki = 1.9 nM T54582 CNT93I 155564947 IC50 = 11.63 nM T54582 C4HEK9 155565565 IC50 = 9.2 nM T54582 CLRN34 155567859 IC50 = 1410 nM T54582 D02VQU 984333 IC50 = 19 nM T83386 D01KKQ 135400182 IC50 = 15 nM T83386 D02LWU 148121 IC50 = 168 nM T83386 D0SV8E 126941 IC50 = 461 nM T83386 D0Y4GO 135410875 IC50 = 42 nM T83386 CPM3L5 67092576 IC50 = 154 nM T83386 CTK64O 67092918 IC50 = 148 nM T83386 C87FBU 135455948 IC50 = 550 nM T83386 CF8D5O 135465664 IC50 > 1000 nM T83386 C9Z4ES 135567027 IC50 = 6.3 nM T83386 C14LTO 135567028 IC50 = 1.82 nM T83386 CF39AI 135567029 IC50 = 0.31 nM T83386 C8N7ES 135567030 IC50 = 2.5 nM T83386 CFE2O7 135567034 IC50 = 0.33 nM T83386 C8KVP5 135567035 IC50 = 0.61 nM T83386 CSQX75 135567163 IC50 = 3.04 nM T83386 CQF8P5 135800109 IC50 = 4.1 nM T83386 CL8VN5 136015502 IC50 = 109 nM T83386 CR7UY3 136044173 IC50 = 9.5 nM T83386 C0Q5FI 136044174 IC50 = 55.7 nM T83386 CGX68Y 136044175 IC50 = 27.4 nM T83386 C4C9FN 136044176 IC50 = 6.6 nM T83386 CIPD35 136044177 IC50 = 661 nM T83386 CZG8W6 136059167 IC50 = 1.3 nM T83386 CZC95Y 136059168 IC50 = 15.02 nM T83386 CG2ID9 136059169 IC50 > 1000 nM T83386 C2WH0S 136059178 IC50 = 186 nM T83386 CB3GL7 136059191 IC50 = 449 nM T83386 CCHG08 136059192 IC50 = 4.43 nM T83386 C4Q1HF 136180345 IC50 = 49.3 nM T83386 CDC83K 136180346 IC50 = 45.5 nM T83386 CF7NW6 136180347 IC50 > 1000 nM T83386 CPH52E 137150145 IC50 > 1000 nM T83386 C9XD1M 137150146 IC50 = 1.78 nM T83386 CHDB56 137150160 IC50 = 1.4 nM T83386 CUF8R1 155515541 IC50 = 1.4 nM T83386 CMKA64 155517044 IC50 = 4.87 nM T83386 CCL3Y9 155518053 IC50 = 0.14 nM T83386 C91SVN 155519837 IC50 = 1.89 nM T83386 CO7BN6 155524531 IC50 > 1000 nM T83386 CT70WU 155530762 IC50 = 0.36 nM T83386 CX42MF 155532591 IC50 = 0.51 nM T83386 CFU98A 155534971 IC50 = 3.01 nM T83386 C4K2RU 155538415 IC50 = 867 nM T83386 C27BIX 155539477 IC50 = 7.78 nM T83386 C6S7OC 155548982 IC50 = 1.12 nM T83386 CX3K8F 155549935 IC50 = 0.58 nM T83386 CJ0MK5 155554671 IC50 = 0.69 nM T83386 CYQ0I9 155555353 IC50 = 1.08 nM T74363 CRTI09 3281693 IC50 = 7000 nM T74363 CMZ3Y7 3281697 IC50 = 10000 nM T74363 C2FV5I 3676137 IC50 = 10000 nM T74363 CAIN92 3676139 IC50 = 5000 nM T74363 C47RMQ 4738040 Ki = 20.8 nM T74363 C4IC9P 5052527 IC50 > 100000 nM T74363 CX7PR4 14449988 Ki = 0.00329 nM T74363 CE2S3V 14449989 Ki = 0.00227 nM T74363 CH09BS 14449992 Ki = 0.00327 nM T74363 CO18RX 15994611 IC50 = 51000 nM T74363 CN73KG 15995634 IC50 = 20000 nM T74363 C13GDN 15995636 IC50 = 36000 nM T74363 CKBP83 16002078 IC50 = 24000 nM T74363 CTW8E4 22421659 IC50 = 21000 nM T74363 C8FVN2 44364233 IC50 > 30000 nM T74363 CZ04YN 44364234 IC50 > 30000 nM T74363 C3O6CP 44364235 IC50 > 30000 nM T74363 C26UCS 44364243 IC50 = 900 nM T74363 C6U1OH 44364244 IC50 = 700 nM T74363 C4U5PA 44364245 IC50 = 80 nM T74363 C61JHV 44364339 IC50 = 50 nM T74363 CWKU04 44364360 IC50 = 60 nM T74363 CA3BD4 44364376 IC50 = 200 nM T74363 CU6L0D 44364420 IC50 = 40 nM T74363 CXR49U 44364421 IC50 > 30000 nM T74363 CU4AE5 44436348 Ki = 500000 nM T74363 C5WE1G 46504414 IC50 = 18000 nM T74363 C35BOE 56589587 Ki = 20000 nM T74363 CIUK84 68295193 IC50 > 100000 nM T74363 C8MDV0 71450599 IC50 = 67000 nM T74363 C4TS3K 71450625 Ki = 0.00217 nM T74363 CT18ZB 71450627 Ki = 0.00636 nM T74363 C9H5UW 71450628 Ki = 0.000589 nM T74363 CE2GY7 71450629 Ki = 0.00653 nM T74363 CO96LQ 71450630 Ki = 0.0044 nM T74363 CLOH40 71452463 Ki = 0.000288 nM T74363 CO0CD2 71452464 Ki = 0.00302 nM T74363 CT8XK3 71454219 Ki = 0.00759 nM T74363 C8JB7E 71455954 IC50 = 30000 nM T74363 CLEN68 71455977 Ki = 0.001 nM T74363 CY36VC 71455978 Ki = 0.011 nM T74363 CIT25C 71457753 IC50 = 146000 nM T74363 C1H8RS 71457776 Ki = 0.0017 nM T74363 CW9IG1 71457777 Ki = 0.0333 nM T74363 CV7EO8 71457778 Ki = 0.012 nM T74363 CLAP24 71459674 IC50 = 30000 nM T74363 C0L4GC 71459695 Ki = 0.00153 nM T74363 CU79DN 71459696 Ki = 0.00445 nM T74363 CTC3X4 71463143 Ki = 0.00411 nM T74363 C2LX6O 92208905 IC50 = 10000 nM T74363 CMSX05 136216669 Ki = 1.33 nM T91331 D03ZBT 11626560 IC50 > 10000 nM T91331 D04LVK 57379345 IC50 = 430 nM T91331 D0H0EQ 24826799 IC50 = 9.4 nM T91331 D00DRL 44137946 IC50 = 50 nM T91331 D02UFQ 11620908 IC50 > 10000 nM T91331 D02WVT 25031915 IC50 = 237.5 nM T91331 D03LWG 53235510 IC50 = 0.7 nM T91331 D05PZB 135398495 IC50 = 10 nM T91331 D07EHV 44814409 IC50 > 10000 nM T91331 D07HPJ 11476171 IC50 > 10000 nM T91331 D0D4VV 46944259 IC50 = 6.4 nM T91331 D0D6XT 118029202 IC50 = 1060 nM T91331 D0E3TC 44259 IC50 = 10.3 nM T91331 D0FD6D 11751922 IC50 = 89 nM T91331 D0H9FR 118295624 Ki = 2.2 nM T91331 D0NW0T 67462786 IC50 = 3 nM T91331 D0VF6E 1401 EC50 = 30 nM T91331 D0XT0W 66555680 IC50 = 22 nM T91331 D03BNU 59604787 IC50 > 10000 nM T91331 D0T3ME 156422 IC50 > 30000 nM T91331 CWH85P 42723 IC50 = 500 nM T91331 CHR70B 237859 IC50 = 120000 nM T91331 C2DG6J 3068873 IC50 = 1400 nM T91331 CPT61U 5328112 IC50 = 290 nM T91331 CDK3J0 5703619 IC50 = 25 nM T91331 CUJR40 10062694 IC50 = 13 nM T91331 CSGD16 10246246 IC50 > 7000 nM T91331 CBOP58 11293798 Ki > 10000 nM T91331 C26BZX 11362471 Ki > 10000 nM T91331 CWXB93 11397177 Ki > 10000 nM T91331 CTG83F 11539329 Ki > 1900 nM T91331 CACS26 11561968 Ki > 2000 nM T91331 CO9KP5 11583459 IC50 > 10000 nM T91331 CMIL86 11590363 Ki > 1900 nM T91331 C69FYK 11604142 Ki = 400 nM T91331 C9T6SC 11640926 Ki > 1900 nM T91331 CU0E8O 11690457 Ki > 2000 nM T91331 CB0AP2 11705863 Ki > 10000 nM T91331 C45EWD 11723489 IC50 > 7000 nM T91331 CFPW41 16007116 Ki > 1900 nM T91331 C9TU1O 16046126 IC50 > 1000 nM T91331 C6JV7W 23400934 IC50 > 7000 nM T91331 CD5S7O 23401001 IC50 > 7000 nM T91331 CWAT04 23630291 IC50 = 7 nM T91331 CMQ6W7 23630305 IC50 = 20 nM T91331 CAJ4T2 24762205 IC50 > 10000 nM T91331 CLBP72 24798571 IC50 > 5741 nM T91331 C6FGQ1 25206346 IC50 = 86 nM T91331 CU9E4P 42629114 IC50 > 10000 nM T91331 CEL61X 44229839 IC50 > 10000 nM T91331 CA98KR 44432441 IC50 > 6000 nM T91331 C6E2SC 45482700 IC50 > 10000 nM T91331 CZXH74 45482750 IC50 > 10000 nM T91331 CUA97D 46209401 IC50 = 280 nM T91331 CY3HW5 46224684 IC50 > 10000 nM T91331 CLS29B 46872626 IC50 > 10000 nM T91331 CHSF07 49806372 IC50 > 1000 nM T91331 C90ANW 50939489 IC50 = 180 nM T91331 CM24LF 52938983 IC50 = 21.5 nM T91331 C09SDH 53257410 IC50 = 4600 nM T91331 C2W9OA 53324451 IC50 > 10000 nM T91331 C4F6SR 53348188 IC50 = 5.99 nM T91331 C8NA4L 53384644 IC50 > 30000 nM T91331 C8AB1J 54759606 Ki = 89 nM T91331 CJN4A5 56594617 IC50 = 505 nM T91331 CV71OR 56594618 IC50 = 125 nM T91331 CM79GX 56594741 IC50 = 66 nM T91331 CMIO24 56594742 IC50 = 115 nM T91331 C2QMD9 56594743 IC50 = 840 nM T91331 CO74WJ 56594744 IC50 = 51 nM T91331 C5G9CR 56594745 IC50 = 54 nM T91331 CHD79F 56594864 IC50 = 9 nM T91331 CMQ2J3 56594865 IC50 = 16 nM T91331 C6FE3Z 56594866 IC50 = 11 nM T91331 CS3E5I 56594867 IC50 = 19 nM T91331 C8P6RD 57505528 IC50 = 4200 nM T91331 CPU2E3 59737752 IC50 = 8000 nM T91331 C1MR8Q 60097495 IC50 > 10000 nM T91331 C9O4GF 66555232 IC50 = 79 nM T91331 CL3EN2 66556938 IC50 = 150 nM T91331 C1HSE0 67035086 IC50 = 2500 nM T91331 CWI6K5 67035106 IC50 > 10000 nM T91331 C38RGB 67035556 IC50 > 10000 nM T91331 CV63UL 67240318 IC50 > 5000 nM T91331 CO6W9D 68004741 IC50 = 3.5 nM T91331 CB6U7F 68005465 IC50 = 4.4 nM T91331 CK83VI 68005486 IC50 = 230 nM T91331 C1RJ7Y 68005600 IC50 = 68 nM T91331 COX3U9 68005621 IC50 = 130 nM T91331 CEXN58 68005732 IC50 = 120 nM T91331 CSK4L6 68208633 IC50 = 12 nM T91331 C8I7GC 68293638 IC50 > 10000 nM T91331 CD56XK 68293660 IC50 > 10000 nM T91331 CEBO91 71452977 IC50 > 10000 nM T91331 CKT60L 71455860 Ki = 1400 nM T91331 CZ31PU 71583657 IC50 > 10000 nM T91331 C9OQ2I 72710839 IC50 = 150 nM T91331 CQ5E3H 73707531 IC50 = 41 nM T91331 CRQO23 86293280 IC50 = 820 nM T91331 C4OC7T 86293469 IC50 = 269 nM T91331 CPG3A5 86302574 IC50 > 30000 nM T91331 CR1N0E 90367910 IC50 = 0.5 nM T91331 CF27DP 91825767 IC50 = 93 nM T91331 CVB8Q7 118728412 IC50 = 71 nM T91331 CH1B5J 118893306 IC50 = 2 nM T91331 C08KEM 122179540 IC50 = 3900 nM T91331 C3AJ4C 122179546 IC50 = 9500 nM T91331 CG0RP7 122179547 IC50 = 4900 nM T91331 C1A0SQ 122179548 IC50 = 5000 nM T91331 C1E4AR 122604567 IC50 > 10000 nM T91331 CY30FL 123752658 IC50 = 1 nM T91331 C9SI5T 127047969 IC50 < 0.2 nM T91331 CUO0C5 132156633 IC50 > 10000 nM T91331 CK9W4F 134135741 IC50 = 7400 nM T91331 CMA60G 134144799 IC50 > 50000 nM T91331 C3MN6B 134144868 IC50 = 4800 nM T91331 CEZH84 134146580 IC50 = 270 nM T91331 C1DF4R 134147544 IC50 = 720 nM T91331 C95NCV 134151662 IC50 = 25 nM T91331 CX7YE1 134155961 IC50 = 18 nM T91331 CE38MW 134156584 IC50 = 4 nM T91331 CVI25K 134157526 IC50 = 940 nM T91331 CO1IL0 134457555 IC50 > 10000 nM T91331 CB15KN 134457556 IC50 > 10000 nM T91331 CCFS35 134457606 IC50 > 10000 nM T91331 CEAH09 134457612 IC50 > 10000 nM T91331 C1P9KY 134457618 IC50 > 10000 nM T91331 CGAV72 134457621 IC50 = 4300 nM T91331 CWZ1L4 135316948 IC50 = 11.6 nM T91331 C5B6XD 135316952 IC50 = 16.3 nM T91331 CWEP52 135316962 IC50 = 7.12 nM T91331 CW5KL0 135316982 IC50 = 12.9 nM T91331 C6E5FP 135317017 IC50 = 5.09 nM T91331 CCTW97 135317286 IC50 = 5.38 nM T91331 CH2JK6 135317468 IC50 = 7.15 nM T91331 CFE0X7 135317546 IC50 = 7.59 nM T91331 C0JM1W 135317567 IC50 = 7.04 nM T91331 CI2L5A 135317791 IC50 = 5.07 nM T91331 CJZ59L 135317844 IC50 = 11.1 nM T91331 C45XNW 135318783 IC50 = 20.5 nM T91331 CLCO61 135398510 IC50 = 3 nM T91331 CS63IO 135476717 IC50 = 108 nM T91331 C4WX3I 135486449 IC50 > 20000 nM T91331 CYXU86 136180312 IC50 = 19580 nM T91331 C9MHA4 136180313 IC50 = 19830 nM T91331 CDT7E4 136211077 IC50 = 2 nM T91331 C7PNC4 136243300 IC50 > 20000 nM T91331 CUN1I4 136243344 IC50 > 20000 nM T91331 C68IKN 136243473 IC50 > 20000 nM T91331 CDY18N 136301774 IC50 = 51000 nM T91331 CH4T8M 136961363 IC50 > 20000 nM T91331 C7N8EG 136961364 IC50 > 20000 nM T91331 CRPQ98 136961365 IC50 > 20000 nM T91331 CSZ16N 136961366 IC50 > 20000 nM T91331 CB9D7F 136961367 IC50 = 19640 nM T91331 CEPT42 136961368 IC50 = 18360 nM T91331 C25ERN 137631967 IC50 = 23 nM T91331 CLQT06 137632162 IC50 > 1000 nM T91331 C0J6IC 137633737 IC50 > 1000 nM T91331 CNX0F9 137634126 IC50 = 40.2 nM T91331 CB35YZ 137634742 IC50 = 560.7 nM T91331 CF7P1V 137635991 IC50 > 1000 nM T91331 C2K8LT 137636345 IC50 > 10000 nM T91331 CUR48O 137636669 IC50 = 3653.5 nM T91331 CF7O2C 137636828 IC50 > 10000 nM T91331 CPR60M 137637024 IC50 > 10000 nM T91331 C06JRX 137637094 IC50 = 122.5 nM T91331 CH2OR6 137637188 IC50 > 1000 nM T91331 CMCI72 137638094 IC50 > 10000 nM T91331 C8AI5O 137638529 IC50 = 430.5 nM T91331 C7J8FB 137639540 IC50 > 10000 nM T91331 CXM2I8 137640932 IC50 = 27.6 nM T91331 CRQG32 137641135 IC50 = 8 nM T91331 C9WBQ0 137641746 IC50 = 279.9 nM T91331 C5E6NQ 137643062 IC50 > 10000 nM T91331 CY8L5M 137644036 IC50 = 150 nM T91331 C0CTB5 137644554 IC50 > 10000 nM T91331 CS3TU7 137644762 IC50 > 10000 nM T91331 C9B7XU 137645188 IC50 = 250.5 nM T91331 CEO3V1 137645361 IC50 > 1000 nM T91331 C09CLU 137646239 IC50 > 1000 nM T91331 C79SUZ 137646264 IC50 = 1200 nM T91331 C7P5AX 137646321 IC50 > 10000 nM T91331 C0YP8D 137646334 IC50 = 22.8 nM T91331 CBK62Y 137646491 IC50 = 93.9 nM T91331 C7CA9N 137646692 IC50 > 10000 nM T91331 CS3H8E 137647913 IC50 > 1000 nM T91331 CGF7X2 137647982 IC50 > 1000 nM T91331 C7EZP8 137649394 IC50 > 10000 nM T91331 CO4HY7 137650511 IC50 = 58.4 nM T91331 CHSB74 137650627 IC50 > 10000 nM T91331 C1DK0P 137651391 IC50 = 15.9 nM T91331 C47VJA 137651444 IC50 = 591.5 nM T91331 CIR94V 137651828 IC50 > 1000 nM T91331 C6EN8I 137652073 IC50 = 35.3 nM T91331 CU5J4G 137652158 IC50 = 969.7 nM T91331 C0MZ1W 137652333 IC50 > 10000 nM T91331 CD7UV3 137652920 IC50 = 401.5 nM T91331 CBAF08 137653174 IC50 > 10000 nM T91331 CTV31U 137653424 IC50 > 1000 nM T91331 CQ85OV 137655810 IC50 > 1000 nM T91331 C01JVI 137656138 IC50 = 388 nM T91331 CV5H3Z 137657932 IC50 = 73.1 nM T91331 C7SEK1 137658232 IC50 > 10000 nM T91331 CQF74K 137658987 IC50 > 10000 nM T91331 C8DZ6L 137659285 IC50 > 10000 nM T91331 C4DT3V 137659387 IC50 > 1000 nM T91331 CY8B6K 137659396 IC50 > 1000 nM T91331 CD3K9G 137659884 IC50 > 1000 nM T91331 C9UMG4 137660300 IC50 > 1000 nM T91331 CS04UY 137660727 IC50 > 1000 nM T91331 CIV31M 137661021 IC50 > 1000 nM T91331 CW9U3A 137661140 IC50 > 10000 nM T91331 C82WHL 137661196 IC50 = 433.8 nM T91331 CM3UF7 137700779 IC50 > 10000 nM T91331 CSRI06 138547901 IC50 = 15 nM T91331 CUXO19 138617501 IC50 = 9.4 nM T91331 C41NGU 138661817 IC50 = 0.41 nM T91331 CZJ5H0 138661862 IC50 = 254.3 nM T91331 C2FSG3 138661878 IC50 = 0.2885 nM T91331 CZD41U 138662420 IC50 = 0.9714 nM T91331 CX9IO0 138662575 IC50 = 0.212 nM T91331 CZ2XH5 139187793 IC50 > 10000 nM T91331 CUH2G6 139554482 IC50 = 1.7 nM T91331 CO9P7G 145351804 IC50 = 10.6 nM T91331 C29XUO 145945978 IC50 = 12.5 nM T91331 C15SAP 145949598 IC50 > 100000 nM T91331 CL14YA 145950580 IC50 > 100000 nM T91331 C1AL5N 145952450 IC50 = 4500 nM T91331 C7MBT6 145957742 IC50 > 100000 nM T91331 CSZ14F 145958261 IC50 > 100000 nM T91331 C93AOR 145980752 IC50 = 3500 nM T91331 CS7TD1 145993995 IC50 > 10000 nM T91331 CN7EF3 145996526 IC50 > 1000 nM T91331 CAQ5R8 154698485 IC50 = 0.3731 nM T91331 C2MD1Q 155513187 IC50 > 10000 nM T91331 C86HPW 155518524 IC50 = 6300 nM T91331 CX37HC 155537699 IC50 > 1000 nM T91331 C35COQ 155538985 IC50 = 330 nM T91331 CYEO53 155555708 IC50 = 6500 nM T91331 D00ERW 44444843 Ki > 1863 nM T91331 D00HVA 11624601 Ki > 1900 nM T91331 D02BXJ 46864270 IC50 = 10.5 nM T91331 D02NNT 53232451 IC50 = 115 nM T91331 D05FFB 91643 IC50 = 400 nM T91331 D06HVH 54613583 IC50 > 10000 nM T91331 D0Q3NG 11715520 Ki > 1900 nM T91331 D0R2WK 16038120 IC50 = 85 nM T91331 D0S7IE 11658882 Ki > 1900 nM T09215 CCK69R 11252976 IC50 = 30900 nM T09215 C2MO4E 56659143 IC50 = 30180 nM T09215 CRZQ62 56662643 IC50 = 36800 nM T09215 C83VOD 56662645 IC50 = 200 nM T09215 C3SUN2 56673013 IC50 = 41210 nM T09215 CD2N5L 56673014 IC50 = 120 nM T09215 CV48HD 56673071 IC50 = 21320 nM T09215 CKP08Y 56676335 IC50 = 1460 nM T09215 CZFK30 56682984 IC50 = 12600 nM T09215 C76FOB 56682985 IC50 = 100 nM T09215 CCA39D 56683043 IC50 = 32460 nM T09215 CUQL27 73346193 IC50 = 142000 nM T09215 CTCP80 73346194 IC50 = 126000 nM T09215 C89JKO 73346195 IC50 = 166000 nM T09215 C35KRO 73346196 IC50 = 190000 nM T09215 C3V2HQ 73347710 IC50 = 156000 nM T09215 C6J2BN 73347711 IC50 = 228000 nM T09215 C0W1YT 73350817 IC50 = 192000 nM T09215 CR3O4M 73353778 IC50 = 172000 nM T09215 C9CZ1M 73353779 IC50 = 208000 nM T09215 CK53DJ 73355301 IC50 = 182000 nM T09215 C19HEM 73355302 IC50 = 204000 nM T09215 CD6J4A 73356848 IC50 = 214000 nM T09215 D0Z1ZI 1678 IC50 = 50700 nM T60606 CDI82V 661788 EC50 = 1160 nM T60606 CUR6Q3 2741928 IC50 > 30000 nM T60606 C79HBK 2887852 EC50 = 5090 nM T60606 C5ROY0 9887381 EC50 = 6500 nM T60606 C5E3TQ 16759579 EC50 = 290 nM T60606 CPJ23F 17757102 EC50 = 930 nM T60606 C9QM7A 17757110 EC50 = 830 nM T60606 CT7ZU9 17757294 EC50 = 3980 nM T60606 CL7X4M 17757296 EC50 = 430 nM T60606 C2LSQ8 17757301 EC50 = 2160 nM T60606 CJWB75 17757314 EC50 = 960 nM T60606 CMK9L4 25246343 EC50 = 90 nM T60606 C53DNJ 25246367 EC50 = 4480 nM T60606 CRXO16 29993669 IC50 > 30000 nM T60606 CY5P9C 29993670 IC50 > 30000 nM T60606 CPZ5S2 46190126 EC50 = 80 nM T60606 C6DI9X 49789101 EC50 = 330 nM T60606 C9U5HB 49789102 EC50 = 1860 nM T60606 CRC4H9 49789103 EC50 = 280 nM T60606 C3TFD2 49789106 EC50 = 2570 nM T60606 C74MXY 49789107 EC50 = 4340 nM T60606 C5XGM3 49789112 EC50 = 18 nM T60606 CVO91Z 49789113 EC50 = 550 nM T60606 CG2NH6 139600336 IC50 = 24000 nM T60606 C0HN5J 139600337 IC50 = 2300 nM T46365 D03GET 4055 IC50 = 2200 nM T46365 D0C0NH 3806 IC50 = 1980 nM T46365 CAD58I 2876 IC50 = 23630 nM T46365 CF1MI3 3136 IC50 = 17400 nM T46365 CI9TK0 3884 IC50 = 42700 nM T46365 C7OJ5H 7013 Ki = 32000 nM T46365 C8JV3A 24465 IC50 = 30000 nM T46365 CB9QR5 39302 IC50 = 23100 nM T46365 CW68ZS 61672 IC50 = 0.93 ug.mL-1 T46365 CF09ZT 71768 IC50 = 12000 nM T46365 C9Z8TW 78723 Ki = 69000 nM T46365 C6G5AH 79441 IC50 = 33100 nM T46365 CQ5T8P 80444 IC50 = 23800 nM T46365 C4S0UL 96582 IC50 = 4600 nM T46365 CFS1T8 133223 Ki = 159000 nM T46365 C2FIH6 149160 IC50 = 4800 nM T46365 CRC4A0 149161 IC50 = 8900 nM T46365 CV9PX7 150081 IC50 = 1500 nM T46365 CXJ37I 231852 Ki = 5300 nM T46365 CT83UE 232961 IC50 = 4130 nM T46365 CK6M9P 233507 IC50 = 12700 nM T46365 C0O2FK 259836 IC50 = 4700 nM T46365 C7H4JI 268982 Ki = 84000 nM T46365 CSH7Q9 272566 IC50 = 4200 nM T46365 CZA6G5 274127 Ki = 80 nM T46365 CKP21I 291456 IC50 = 7900 nM T46365 C13WRN 315113 IC50 = 20100 nM T46365 CV6AX0 320851 IC50 = 1600 nM T46365 C05EMO 351827 IC50 = 250 nM T46365 CI3K5N 378911 IC50 = 900 nM T46365 C7BAY8 379075 IC50 = 930 nM T46365 C5Q7BU 386231 IC50 = 510 nM T46365 C02WIT 388306 IC50 = 3000 nM T46365 C75COU 470952 IC50 = 4900 nM T46365 CO4J7N 470958 IC50 = 24300 nM T46365 CYZI40 604273 IC50 > 50000 nM T46365 CH35LS 662869 IC50 = 2000 nM T46365 C1DH0C 674157 IC50 = 5300 nM T46365 CDI2W3 719031 IC50 = 10900 nM T46365 C2B6EK 752982 IC50 = 16000 nM T46365 C5MQP8 852158 IC50 > 100000 nM T46365 C6OSR1 914570 IC50 = 9100 nM T46365 CI87JW 1001784 IC50 = 2690 nM T46365 C6IW2P 1131425 IC50 = 19000 nM T46365 C9K1SE 1177946 IC50 = 6000 nM T46365 CM23EO 1239196 IC50 = 37400 nM T46365 CFR61E 1307198 IC50 = 5900 nM T46365 CQW6F7 1308005 IC50 = 900 nM T46365 C9VW4Y 1332846 IC50 = 5400 nM T46365 CKD92S 1383304 IC50 = 1980 nM T46365 C3VIK9 1398345 IC50 = 4670 nM T46365 C91NQB 1400320 IC50 = 2500 nM T46365 CSC9W6 1400627 IC50 = 1700 nM T46365 CH3M0Z 1401217 IC50 = 4700 nM T46365 C4U8DM 1413573 IC50 = 1600 nM T46365 C8J2ZI 1864385 IC50 = 4400 nM T46365 C7M4ID 1895639 IC50 = 5000 nM T46365 CU0A3X 1921859 IC50 = 200 nM T46365 C9CS3K 1925936 IC50 = 10900 nM T46365 C4RH2W 1933357 IC50 = 210 nM T46365 CRFK64 1953519 IC50 = 8600 nM T46365 C9JQ2O 1968455 IC50 = 4200 nM T46365 C6N7ZI 2142225 IC50 = 3300 nM T46365 C7NJB6 2323972 IC50 = 830 nM T46365 CO9ST2 2446135 IC50 = 13600 nM T46365 CF5BV8 2734086 IC50 = 23230 nM T46365 COE91V 2742421 IC50 = 3100 nM T46365 C7JO4Q 2820003 IC50 = 1700 nM T46365 C7SBI5 2894962 IC50 = 31900 nM T46365 C5AZL4 2941397 IC50 = 13700 nM T46365 CWK5N4 3281033 IC50 = 3370 nM T46365 C5D1CR 4194417 IC50 > 50000 nM T46365 CYN3Z9 4263321 IC50 = 11100 nM T46365 C6R3WL 4343361 IC50 = 9100 nM T46365 CRH60Z 4460044 IC50 = 10750 nM T46365 C2LC1E 5130755 IC50 = 770 nM T46365 CWIC65 5279637 IC50 = 5200 nM T46365 C8CTS9 5279656 IC50 = 1000 nM T46365 CK8ZM5 5336010 IC50 = 13000 nM T46365 C5IC3F 5461522 IC50 = 300 nM T46365 C4VM8J 9173830 IC50 = 14900 nM T46365 CP3AO9 9356353 IC50 = 17500 nM T46365 CZ93IR 9356454 IC50 = 10100 nM T46365 CF79QB 9421427 IC50 = 22700 nM T46365 CIAT52 9865848 IC50 = 19000 nM T46365 C30KRC 9896432 IC50 = 100000 nM T46365 C3MUO6 9903359 IC50 = 6500 nM T46365 C0CJ7U 9926573 IC50 = 5900 nM T46365 CRU8E0 9978702 IC50 = 1620 nM T46365 COU6V1 9978703 IC50 = 1880 nM T46365 COB58D 10092773 IC50 = 1900 nM T46365 CEJN86 10253374 Ki = 4600 nM T46365 CUD28W 10318951 IC50 = 18000 nM T46365 CYX58O 10350397 IC50 = 15000 nM T46365 C5RFM3 10411670 IC50 = 3400 nM T46365 C05SVE 10444314 IC50 = 3000 nM T46365 C4HE0C 10458201 IC50 = 25000 nM T46365 C2B8AM 10476452 IC50 = 1440 nM T46365 CY93MH 10513846 IC50 = 9520 nM T46365 C5A3WY 11200445 IC50 = 10000 nM T46365 CXN1S5 11269661 IC50 = 87000 nM T46365 CQJ07W 11299775 IC50 > 100000 nM T46365 CU4E2B 11391905 IC50 > 100000 nM T46365 CRPL64 11516963 IC50 = 16100 nM T46365 C1M2NH 11576677 IC50 = 2000 nM T46365 C4ANG0 12166238 Ki = 22000 nM T46365 C2PU6E 12227519 IC50 = 850 nM T46365 CD3K8H 12387018 IC50 = 28800 nM T46365 CP8FX1 12824032 IC50 = 14200 nM T46365 CSC25V 14149682 IC50 = 55200 nM T46365 CY3JU7 14646108 IC50 > 100000 nM T46365 CDJP28 15322751 IC50 = 1950 nM T46365 CU8J6A 16126459 IC50 = 7600 nM T46365 C8CSM3 16126550 IC50 = 8700 nM T46365 C29ZMK 16126551 IC50 = 11600 nM T46365 C3TPL7 16126552 IC50 = 3600 nM T46365 CETU13 16727376 IC50 = 1160 nM T46365 C94XRY 16727378 IC50 = 13630 nM T46365 CP10YE 16727381 IC50 = 3310 nM T46365 C7X6FT 16727382 IC50 = 1210 nM T46365 CC01XD 16727384 IC50 = 1850 nM T46365 CJ6DA4 16727385 IC50 = 4190 nM T46365 C7OJN8 16727387 IC50 = 2570 nM T46365 CW3BF9 16727388 IC50 = 5250 nM T46365 C4Z6BF 17483715 IC50 = 8900 nM T46365 C04GYC 17531735 IC50 = 19000 nM T46365 CX42CP 17554676 IC50 = 12100 nM T46365 CFU3D7 18350018 IC50 = 4550 nM T46365 CWF29X 21190797 Ki = 30000 nM T46365 C5O0SV 24204784 Ki = 4700 nM T46365 CE9B6H 25014222 IC50 = 3920 nM T46365 CT5AV2 25147777 IC50 = 14160 nM T46365 C6NR5D 44249868 IC50 = 2300 nM T46365 CPK9I3 44290909 IC50 = 11000 nM T46365 CDZ5E4 44290922 IC50 > 30000 nM T46365 CET01O 44291005 IC50 > 30000 nM T46365 C4DLS2 44291008 IC50 = 8700 nM T46365 CB1N0Q 44291022 IC50 = 6500 nM T46365 CO20QR 44291106 IC50 = 4900 nM T46365 CGF21I 44291115 IC50 > 30000 nM T46365 C1VW4N 44291292 IC50 = 3500 nM T46365 C3NT7L 44291345 IC50 > 30000 nM T46365 CQ6B3L 44291358 IC50 = 11000 nM T46365 C72MBY 44291368 IC50 = 29000 nM T46365 CM4IY6 44291369 IC50 > 30000 nM T46365 C9VPG5 44291386 IC50 > 30000 nM T46365 CTG6D5 44291394 IC50 = 4900 nM T46365 CP9S0X 44291405 IC50 > 30000 nM T46365 CK4VB3 44291414 IC50 = 7800 nM T46365 C67CXQ 44291439 IC50 > 30000 nM T46365 CMZ48B 44291450 IC50 > 30000 nM T46365 C97MYZ 44291451 IC50 > 30000 nM T46365 CDT1U4 44291454 IC50 > 30000 nM T46365 C7B0PO 44291526 IC50 = 8400 nM T46365 C1O4DS 44291543 IC50 = 11000 nM T46365 CVI05R 44291544 IC50 = 9300 nM T46365 CJ4B9F 44291668 IC50 = 7100 nM T46365 CFK34Q 44291735 IC50 > 30000 nM T46365 CE13LX 44291762 IC50 = 7900 nM T46365 CGNM73 44291786 IC50 = 5600 nM T46365 CED95K 44291814 IC50 = 8500 nM T46365 CK7LP3 44291815 IC50 = 7500 nM T46365 CDJ1S7 44301133 IC50 = 2130 nM T46365 C7YN6L 44318744 IC50 > 2000000 nM T46365 CK69BS 44320206 IC50 = 27000 nM T46365 CD9Z6B 44320207 IC50 > 300000 nM T46365 CM17GK 44337392 IC50 = 72000 nM T46365 CXJO75 44337399 IC50 = 20000 nM T46365 CQV1I5 44337400 IC50 = 80000 nM T46365 CZQ8F0 44337401 IC50 = 14000 nM T46365 CZ79HK 44337402 IC50 > 100000 nM T46365 C75MSY 44337409 IC50 > 100000 nM T46365 CUD0O4 44337410 IC50 = 89000 nM T46365 C84VJN 44337423 IC50 = 33000 nM T46365 CQ3F5T 44337439 IC50 = 46000 nM T46365 CQN51Y 44337440 IC50 = 69000 nM T46365 C7X2CV 44337441 IC50 > 100000 nM T46365 C91ALN 44337454 IC50 = 92000 nM T46365 CTVW60 44337518 IC50 = 38000 nM T46365 CLW6G3 44337519 IC50 = 34000 nM T46365 C78WUC 44337562 IC50 = 89000 nM T46365 CRT7I6 44337574 IC50 = 54000 nM T46365 C5A9TD 44337575 IC50 > 100000 nM T46365 C7S3VN 44337581 IC50 = 76000 nM T46365 CC1K8N 44337589 IC50 = 58000 nM T46365 C6K3MN 44337596 IC50 = 88000 nM T46365 CG4X5N 44337597 IC50 = 70000 nM T46365 C6YJ9T 44337604 IC50 = 26000 nM T46365 CM6NJ2 44337607 IC50 > 100000 nM T46365 C90YQX 44337608 IC50 = 21000 nM T46365 C9VCW0 44337612 IC50 > 100000 nM T46365 C1OW4N 44337711 IC50 = 26000 nM T46365 CVW17B 44337712 IC50 = 22000 nM T46365 CD06ZI 44337719 IC50 = 40000 nM T46365 CXRJ74 44337726 IC50 > 100000 nM T46365 CNZ12Q 44337727 IC50 = 33000 nM T46365 C0I5NO 44337786 IC50 = 34000 nM T46365 CTRH27 44337799 IC50 > 100000 nM T46365 CV6U7P 44337816 IC50 > 100000 nM T46365 CTM46P 44372707 IC50 = 70000 nM T46365 CF76EN 44372708 IC50 = 100000 nM T46365 CHU1F9 44372735 IC50 = 70000 nM T46365 CC9F1R 44372757 IC50 = 27000 nM T46365 CFXB91 44372784 IC50 = 33000 nM T46365 C1B0AJ 44372916 IC50 = 90000 nM T46365 CC2SP9 44372918 IC50 = 90000 nM T46365 COJ45R 44372927 IC50 = 50000 nM T46365 CSUP53 44372935 IC50 = 36000 nM T46365 C5LF3J 44372958 IC50 = 50000 nM T46365 CS9P1D 44372965 IC50 = 90000 nM T46365 CA46ZJ 44372969 IC50 = 27000 nM T46365 CS5OU3 44372970 IC50 = 60000 nM T46365 CQ04HO 44372974 IC50 = 35000 nM T46365 CH9AD7 44372994 IC50 = 32000 nM T46365 CXS37O 44373002 IC50 = 75000 nM T46365 C3ALC1 44373005 IC50 = 27000 nM T46365 C70HLK 44373008 IC50 = 52000 nM T46365 C3WDB1 44373034 IC50 = 30000 nM T46365 CPK29B 44373043 IC50 = 35000 nM T46365 CO21LB 44373045 IC50 > 100000 nM T46365 CP0J7V 44373047 IC50 = 40000 nM T46365 C9X1BL 44373062 IC50 = 45000 nM T46365 CV76QK 44373065 IC50 > 100000 nM T46365 CJ9W0B 44373081 IC50 = 75000 nM T46365 CWO35H 44373086 IC50 = 45000 nM T46365 CR2A1O 44373117 IC50 = 30000 nM T46365 C0JS5Z 44373134 IC50 = 30000 nM T46365 CJ18HL 44373160 IC50 = 35000 nM T46365 CC1ZI8 44373161 IC50 = 59000 nM T46365 C0AL4K 44373187 IC50 = 90000 nM T46365 CLHR95 44373202 IC50 = 58000 nM T46365 CAF0D1 44373220 IC50 = 45000 nM T46365 C6RCE2 44373226 IC50 = 75000 nM T46365 C5CP8D 44373228 IC50 = 55000 nM T46365 CRW3C6 44373229 IC50 = 55000 nM T46365 C70OGF 44373231 IC50 = 30000 nM T46365 C03QOL 44373233 IC50 = 45000 nM T46365 CO7CH3 44373234 IC50 = 50000 nM T46365 CD21NJ 44373243 IC50 = 35000 nM T46365 C19VAQ 44373247 IC50 = 57000 nM T46365 C5K4EP 44373278 IC50 = 33000 nM T46365 C9JOA3 44373294 IC50 = 40000 nM T46365 CQZ15M 44373295 IC50 = 36000 nM T46365 CO34TQ 44373296 IC50 = 40000 nM T46365 C0LVW5 44373304 IC50 = 62000 nM T46365 CM7FO8 44373314 IC50 = 75000 nM T46365 CZ16HA 44373332 IC50 = 60000 nM T46365 C8LVK4 44373346 IC50 = 80000 nM T46365 C63AFP 44373356 IC50 = 20000 nM T46365 C90HPA 44373357 IC50 = 55000 nM T46365 C94ZPN 44373371 IC50 = 45000 nM T46365 CXY12L 44373385 IC50 = 40000 nM T46365 CZG9H8 44373386 IC50 = 50000 nM T46365 CKR6Q7 44373395 IC50 = 70000 nM T46365 CT1IO5 44373398 IC50 = 35000 nM T46365 C8OGM9 44373404 IC50 = 30000 nM T46365 CPR19J 44373405 IC50 = 66000 nM T46365 C09AUB 44373407 IC50 = 45000 nM T46365 C01FXG 44373444 IC50 = 23000 nM T46365 C3ERO7 44373445 IC50 = 23000 nM T46365 CNY95Z 44373455 IC50 = 28000 nM T46365 CTQX83 44373644 IC50 = 15000 nM T46365 CFL91W 44392831 IC50 = 5800 nM T46365 C54CFD 44392873 IC50 = 5000 nM T46365 CX28MD 44406938 IC50 = 120 nM T46365 C4VO7S 44407055 IC50 = 10000 nM T46365 CYW68I 44409605 IC50 = 7550 nM T46365 CGX23J 44409674 IC50 = 3780 nM T46365 CTM56S 44409675 IC50 = 3630 nM T46365 C6E4UN 44409680 IC50 = 2580 nM T46365 C25MUW 44409681 IC50 = 3160 nM T46365 CTL17C 44409833 IC50 = 13820 nM T46365 CB31QM 44409834 IC50 = 3990 nM T46365 CY6QB9 44409856 IC50 = 4850 nM T46365 C23ERY 44409919 IC50 = 5330 nM T46365 CB96NM 44409921 IC50 = 7540 nM T46365 C56DNZ 44409999 IC50 = 5070 nM T46365 CH08EI 44410004 IC50 = 4090 nM T46365 C94QYM 44410005 IC50 = 4630 nM T46365 C0S8RA 44424744 IC50 = 47700 nM T46365 C9SJ3O 44424745 IC50 = 6700 nM T46365 C7LJB2 44579573 IC50 = 11200 nM T46365 C09QYC 44579574 IC50 = 10000 nM T46365 COUG36 44579618 IC50 = 1750 nM T46365 CQ7V2Z 44579619 IC50 = 3400 nM T46365 CLIK47 45267539 IC50 = 2600 nM T46365 C3IQM0 45267545 IC50 = 5200 nM T46365 C2MDQ6 45270955 IC50 = 6900 nM T46365 CCG19S 45922965 IC50 = 20100 nM T46365 C7ZS4V 46218884 IC50 = 7800 nM T46365 C81CPM 46861833 IC50 = 160 nM T46365 C0A9LD 46861834 IC50 = 120 nM T46365 C0OHS1 46887676 IC50 = 3360 nM T46365 CW3I9Y 46887819 IC50 = 1390 nM T46365 CPK9Y1 46887820 IC50 = 500 nM T46365 C5ZI4N 46887821 IC50 = 400 nM T46365 CL98EV 46887869 IC50 = 1110 nM T46365 CRVH84 46887870 IC50 = 450 nM T46365 CAO6I7 46887871 IC50 = 1470 nM T46365 CYZ9O2 46887872 IC50 = 540 nM T46365 C2NKS5 46887901 IC50 = 240 nM T46365 CG3OX4 46887902 IC50 = 170 nM T46365 CT0Z5F 46887903 IC50 = 250 nM T46365 CHW0N4 46888132 IC50 = 1010 nM T46365 CM46ER 46888133 IC50 = 960 nM T46365 CGS1I2 46888134 IC50 = 520 nM T46365 C9AD3E 46888135 IC50 = 540 nM T46365 CPEG29 46888174 IC50 = 230 nM T46365 CLD8H9 46888175 IC50 = 2130 nM T46365 CHRJ95 46888176 IC50 = 2600 nM T46365 CUN8E6 46888177 IC50 = 4330 nM T46365 C6YCR9 46888226 IC50 = 410 nM T46365 CY37BH 46888227 IC50 = 490 nM T46365 C0RI2C 46888228 IC50 = 320 nM T46365 CXYT94 46888285 IC50 = 1150 nM T46365 CP15RA 46888286 IC50 = 730 nM T46365 CVLX06 46888287 IC50 = 2080 nM T46365 CGF9R5 46888288 IC50 = 340 nM T46365 C8X0GZ 46888360 IC50 = 2920 nM T46365 CO81MP 46888361 IC50 = 310 nM T46365 C84ZYT 46888362 IC50 = 30000 nM T46365 COD47H 46888363 IC50 = 5080 nM T46365 CMDB84 53316640 IC50 = 25400 nM T46365 C9GVU5 53317937 IC50 = 43300 nM T46365 CV4QD5 53317938 IC50 = 9900 nM T46365 CWT10N 53319270 IC50 > 50000 nM T46365 CRC82E 53320578 IC50 = 38200 nM T46365 C8Y4KW 53320579 IC50 = 3900 nM T46365 CF35GK 53320580 IC50 = 7000 nM T46365 C04CYS 53320581 IC50 > 50000 nM T46365 CBI29Z 53321875 IC50 = 11900 nM T46365 C94WKB 53324565 IC50 = 39700 nM T46365 C4N1OE 53763809 Ki = 54000 nM T46365 CCNG89 54576098 IC50 = 4580 nM T46365 CV3YH5 54576318 IC50 = 5130 nM T46365 C4CAU1 54576319 IC50 = 3080 nM T46365 CYK80P 54576320 IC50 = 2630 nM T46365 CKD3W9 54576321 IC50 = 2890 nM T46365 C1P4QM 54576322 IC50 = 2490 nM T46365 CIE87V 54585167 IC50 = 1900 nM T46365 CE94WN 54587113 IC50 = 50000 nM T46365 CQ30US 54685915 IC50 = 12400 nM T46365 CZ82GO 54695794 IC50 > 100000 nM T46365 CT7S1R 54697955 IC50 = 13700 nM T46365 CW3M8N 54706178 IC50 > 100000 nM T46365 C73TSH 54718593 IC50 = 8000 nM T46365 CB96GH 54768270 IC50 = 19380 nM T46365 C1GDN4 54768308 IC50 = 8440 nM T46365 CM8H3X 54768309 IC50 = 13730 nM T46365 CB80UX 54768349 IC50 = 15180 nM T46365 C2R5JW 54768350 IC50 = 14680 nM T46365 C1VCJ9 54768351 IC50 = 6600 nM T46365 CF7X2K 54768352 IC50 = 5350 nM T46365 C48KOI 54768353 IC50 = 8930 nM T46365 CK3W0Z 54768391 IC50 = 5630 nM T46365 C01LRT 54768392 IC50 = 10740 nM T46365 C8DLG4 54768393 IC50 = 14030 nM T46365 CPGC13 54768394 IC50 = 7040 nM T46365 CVA04X 54768395 IC50 = 11640 nM T46365 CHM5V3 56660070 IC50 = 67500 nM T46365 CHOF39 56670422 IC50 = 8200 nM T46365 CI9R8M 56670423 IC50 > 120000 nM T46365 CL3N0K 56673907 IC50 = 27100 nM T46365 CAL96I 56673908 IC50 = 11600 nM T46365 CEK3S2 56680547 IC50 = 20600 nM T46365 CN3EW7 56683882 IC50 = 31100 nM T46365 C5CQY2 56683883 IC50 = 12200 nM T46365 CV4PW2 56683884 IC50 = 6200 nM T46365 CZP28F 57327772 IC50 = 11300 nM T46365 CO2F6B 57327843 IC50 = 17100 nM T46365 CIQP45 57327844 IC50 = 13810 nM T46365 C1N9XS 57327846 IC50 = 28150 nM T46365 C79IOT 57327917 IC50 = 10900 nM T46365 CVFR71 58978690 Ki = 7100 nM T46365 CWBE16 66525293 IC50 = 23700 nM T46365 CZ8ID6 66848959 IC50 = 5900 nM T46365 CHUI31 69188146 Ki = 6100 nM T46365 CP10SK 70240311 IC50 = 10800 nM T46365 C7VES4 71449486 IC50 = 13720 nM T46365 CY07HW 71456616 IC50 = 6120 nM T46365 C4N3CF 71496104 IC50 = 1660000 nM T46365 CMAI62 71496106 IC50 = 2740000 nM T46365 CY1CH5 71496217 IC50 = 3660000 nM T46365 CWJ2O7 71496218 IC50 = 3390000 nM T46365 CTU0X5 71496219 IC50 = 2870000 nM T46365 C2H3ZC 71511772 IC50 = 2470000 nM T46365 CJ2ZQ7 71697056 IC50 = 14400 nM T46365 C6PFD1 73345215 IC50 = 3300 nM T46365 CGC60U 73346748 IC50 = 1700 nM T46365 CHBJ65 73346749 IC50 = 1200 nM T46365 C5DV3I 73346750 IC50 = 3000 nM T46365 C5PYT7 73349825 IC50 = 4500 nM T46365 C3QPK5 73349826 IC50 = 1300 nM T46365 C3WGM7 73351344 IC50 = 3700 nM T46365 C1DWU4 73353952 IC50 = 7370 nM T46365 C9UP3V 73353954 IC50 = 1620 nM T46365 C15NCG 73354312 IC50 = 6800 nM T46365 CS5O4J 73355491 IC50 = 2510 nM T46365 CMDC47 73357035 IC50 = 4940 nM T46365 CY0K7L 73357036 IC50 = 9740 nM T46365 CS76KU 90666197 IC50 = 3500 nM T46365 C96RMI 90666198 IC50 = 4200 nM T46365 C1Y9EK 90666199 IC50 = 6800 nM T46365 CZ50TY 90666200 IC50 = 19700 nM T46365 CP94DI 90666344 IC50 = 2190 nM T46365 CBK96X 90666455 IC50 = 3380 nM T46365 C61PBQ 90666456 IC50 = 2400 nM T46365 C40WCO 90666457 IC50 = 5410 nM T46365 C2ZGE9 90666458 IC50 = 2830 nM T46365 CG5TY1 90666459 IC50 = 4880 nM T46365 CWQN87 90666460 IC50 = 3660 nM T46365 CLU52N 90666461 IC50 = 4820 nM T46365 C0DW7A 90666462 IC50 = 2550 nM T46365 CXMC74 90666463 IC50 = 4380 nM T46365 C1WY6D 101738247 Ki = 6500 nM T46365 C0WNF2 118710330 IC50 = 1.24 ug.mL-1 T46365 CY8D7B 118710331 IC50 = 4.07 ug.mL-1 T46365 CH8TQ0 118710335 IC50 = 3.26 ug.mL-1 T46365 CFT67U 118710337 IC50 = 4.46 ug.mL-1 T46365 CM79HY 118710338 IC50 = 4.59 ug.mL-1 T46365 CQ1TN4 118710342 IC50 = 3.96 ug.mL-1 T46365 C7ZLK3 118710343 IC50 = 2.63 ug.mL-1 T46365 C47QMJ 118710344 IC50 = 3.36 ug.mL-1 T46365 CN2XA6 118710346 IC50 = 2.49 ug.mL-1 T46365 CX89NJ 118710347 IC50 = 3.11 ug.mL-1 T46365 CUG17X 118710348 IC50 = 1.18 ug.mL-1 T46365 CH38YV 118710350 IC50 = 4.11 ug.mL-1 T46365 C87BLJ 118710352 IC50 = 2.21 ug.mL-1 T46365 C83ZLF 118710354 IC50 = 2.21 ug.mL-1 T46365 CPJ98Q 118710355 IC50 = 2.61 ug.mL-1 T46365 CPS0R7 118710356 IC50 = 8.01 ug.mL-1 T46365 CP5NK7 118710357 IC50 = 1.28 ug.mL-1 T46365 CIQ1S5 118710358 IC50 = 4.78 ug.mL-1 T46365 CUD6A9 118710359 IC50 = 1.57 ug.mL-1 T46365 C9SH1O 118710360 IC50 = 3 ug.mL-1 T46365 C36KIZ 118721518 IC50 = 42920 nM T46365 CI65JN 118737609 IC50 = 6300 nM T46365 C82KRX 118737610 IC50 > 100000 nM T46365 CC2ZT6 118737611 IC50 = 7200 nM T46365 CY6K0I 118737612 IC50 = 13600 nM T46365 CB0CS9 118737613 IC50 = 6500 nM T46365 CE4RH2 118737614 IC50 = 5500 nM T46365 CA1VM7 118737695 IC50 = 4600 nM T46365 CU6SD1 118737696 IC50 = 7000 nM T46365 CM92PW 121344571 IC50 <= 9000 nM T46365 CRFQ07 124165614 Ki = 2800 nM T46365 C71BDH 134132879 IC50 = 5830000 nM T46365 C6DCR0 135420883 IC50 = 2600 nM T46365 CBD5C3 135420929 IC50 = 2300 nM T46365 CS1KZ3 135441149 IC50 = 4500 nM T46365 C0P6TV 135444298 IC50 = 3200 nM T46365 CG2Q6N 135444322 IC50 = 3700 nM T46365 C9NYV1 135444837 IC50 = 8900 nM T46365 CW3L5Z 135451595 IC50 = 9900 nM T46365 CRV42A 135451647 IC50 = 2100 nM T46365 C2I3NM 135458252 IC50 = 2300 nM T46365 CX9AV5 135469884 IC50 = 1800 nM T46365 C04TVF 135512954 IC50 = 2100 nM T46365 CV1ZB2 135522709 IC50 = 2800 nM T46365 C78BVZ 135527488 IC50 = 2700 nM T46365 CJRX49 135529547 IC50 = 4400 nM T46365 CF8V7A 135529575 IC50 = 3100 nM T46365 CDP6X2 135629644 IC50 = 1200 nM T46365 CCMG69 135658050 IC50 = 2300 nM T46365 CO06BL 135665679 IC50 = 3300 nM T46365 CSC48W 135700427 IC50 = 3900 nM T46365 C2V7NL 135797380 IC50 = 6550 nM T46365 C27EYJ 135797381 IC50 = 3150 nM T46365 CZOL36 135797386 IC50 = 8610 nM T46365 CBX75S 135797387 IC50 > 100000 nM T46365 C2L6UZ 135797388 IC50 = 3330 nM T46365 C0S1VO 135797389 IC50 = 8310 nM T46365 CS40TI 135797392 IC50 > 100000 nM T46365 C0RJW6 135797397 IC50 = 4230 nM T46365 C5UL0V 135955126 IC50 = 8420 nM T46365 C9YRO4 135966042 IC50 = 5100 nM T46365 C85VGD 136069445 IC50 = 4260 nM T46365 C49POR 136216675 IC50 = 1380 nM T46365 CJA8P0 136216676 IC50 = 3400 nM T46365 CTX10A 136216677 IC50 = 11900 nM T46365 C50MCG 136216678 IC50 = 2500 nM T46365 CY73XR 136216679 IC50 = 13900 nM T46365 CP3QE4 136216680 IC50 = 21000 nM T46365 C96JZW 136216681 IC50 = 2700 nM T46365 CEWV20 136216682 IC50 = 2200 nM T46365 CHD0M4 136216683 IC50 = 7500 nM T46365 C25EAK 136216684 IC50 = 6600 nM T46365 CUQ4C9 136216685 IC50 = 3900 nM T46365 CL7N1J 136216686 IC50 = 3500 nM T46365 CY5N1D 136216687 IC50 = 8400 nM T46365 CW70QB 136216688 IC50 = 2900 nM T46365 C1NO6Y 136216689 IC50 = 8500 nM T46365 CFZ57E 136216690 IC50 = 57300 nM T46365 CHB7P6 136216691 IC50 = 4400 nM T46365 CG1E2F 136216692 IC50 = 2900 nM T46365 C43NXE 136216693 IC50 = 2400 nM T46365 CTD81Y 136216694 IC50 = 7700 nM T46365 C76EGN 136216695 IC50 = 13800 nM T46365 C74AVN 136216696 IC50 = 11200 nM T46365 C69ZKV 136216697 IC50 = 20600 nM T46365 C23ZHC 136216698 IC50 = 40100 nM T46365 CNEJ36 136216699 IC50 = 48400 nM T46365 CQ7L2H 136254273 IC50 = 5520 nM T46365 C5C1XF 136254274 IC50 = 13100 nM T46365 CL4A5E 136254275 IC50 = 23800 nM T46365 CH7N3Z 136254276 IC50 = 6230 nM T46365 CL4ZM7 136254277 IC50 = 13500 nM T46365 CAHC90 136254278 IC50 = 7530 nM T46365 CQ84LN 136254279 IC50 = 12100 nM T46365 CBEU97 136254280 IC50 = 5750 nM T46365 C3LK1C 136254281 IC50 = 5130 nM T46365 CNMJ89 138911333 Ki = 8500 nM T46365 CB2D3K 139600304 IC50 = 1390 nM T46365 CIN0D1 145964209 IC50 = 8400 nM T46365 CA7G2L 145966685 IC50 = 17300 nM T46365 C7EQ9U 145978118 IC50 = 6700 nM T46365 CW36SM 145978264 IC50 = 22500 nM T46365 CW9CN5 155512425 Ki = 34000 nM T46365 CT61BM 155512612 Ki = 2900 nM T46365 C2C4FI 155512986 Ki = 800 nM T46365 CC67QM 155513419 Ki = 1400 nM T46365 CO96DC 155513532 Ki = 45000 nM T46365 CE4G3Y 155516097 Ki = 5100 nM T46365 CGUP05 155517773 IC50 = 380 nM T46365 CPM65J 155520600 Ki = 11900 nM T46365 CZ75SL 155521073 IC50 = 490 nM T46365 CER17A 155530495 Ki = 9900 nM T46365 C0HV8I 155531212 Ki = 36000 nM T46365 CZ3FY0 155531253 Ki = 5800 nM T46365 CCQ48F 155531806 IC50 = 2790 nM T46365 C9A1KU 155535895 Ki = 36000 nM T46365 CTHD18 155536274 Ki = 6900 nM T46365 CQ63GA 155537698 IC50 = 320 nM T46365 CRU6F2 155538623 IC50 = 830 nM T46365 C8D4BZ 155538725 Ki = 4900 nM T46365 C5NI4P 155541989 Ki = 7300 nM T46365 C25DOA 155543411 Ki = 55000 nM T46365 CF2J7D 155543449 Ki = 7400 nM T46365 C4D5MV 155543902 IC50 = 1000 nM T46365 CAB15R 155555347 Ki = 12500 nM T46365 C3D2FE 155556249 Ki = 16900 nM T46365 CY6UM8 155557874 Ki = 6400 nM T46365 C9ZMO5 155566711 Ki = 2700 nM T46365 CU3F9X 155569214 Ki = 13400 nM T46365 D00SAA 14828129 IC50 = 24100 nM T46365 D02UHP 255964 IC50 = 5300 nM T46365 D04OXY 16871 IC50 = 46800 nM T46365 D07JRA 44409685 IC50 = 3230 nM T46365 D07REK 343759 IC50 = 270 nM T46365 D08GWQ 44409669 IC50 = 10860 nM T46365 D0AS0V 10141 IC50 = 1000 nM T46365 D0DQ6Z 8530 IC50 = 2760 nM T46365 D0J1KH 262093 IC50 = 100 nM T46365 D0L5LN 6780 IC50 = 9510 nM T46365 D0M2EM 4650 IC50 > 50000 nM T46365 D0N7YT 44409922 IC50 = 4530 nM T46365 D0P0IE 10205 IC50 = 3100 nM T46365 D0SI7S 44582382 IC50 = 9530 nM T46365 D0SJ2Q 10494 IC50 = 980 nM T46365 D0X5WD 44409841 IC50 = 8710 nM T92609 D00JVR 2267 Ki = 50.12 nM T92609 D01AZG 5073 Ki = 2.8 nM T92609 D01JUF 5775 Ki = 0.6 nM T92609 D03MIR 3157 Ki = 0.537 nM T92609 D03SKR 2803 Ki = 512.86 nM T92609 D04DKH 4418 Ki = 3.7 nM T92609 D04JEE 4946 EC50 > 5011.87 nM T92609 D04PHC 5816 EC50 = 400 nM T92609 D05MBZ 129211 Ki = 0.029 nM T92609 D05ZIK 4205 IC50 = 3162.28 nM T92609 D06OFS 68712 Ki = 6025.6 nM T92609 D07MOX 439260 EC50 = 9.1 nM T92609 D08JIV 2162 Ki = 2344 nM T92609 D09EBS 4636 Ki = 15.85 nM T92609 D09GYT 6082 EC50 = 720 nM T92609 D09MWJ 2092 Ki = 8.2 nM T92609 D0AE3X 2435 Ki = 2818.38 nM T92609 D0G8NN 119570 Ki > 10000 nM T92609 D0H3HM 60795 Ki = 100 nM T92609 D0H4JM 8969 Ki = 1057 nM T92609 D0H7KF 5002 Ki = 100 nM T92609 D0O6IU 6041 EC50 = 55 nM T92609 D0O6IZ 4436 EC50 = 63.1 nM T92609 D0P9RF 5401 Ki = 2 nM T92609 D0R6RO 4184 IC50 = 407.38 nM T92609 D0U0VU 5312125 Ki = 0.036 nM T92609 D0V4QS 135398745 Ki = 60 nM T92609 D0WV3U 4893 Ki = 0.04 nM T92609 D0Y4DY 5709 Ki = 91 nM T92609 D0Z1RV 135398737 Ki = 10 nM T92609 D0LI1C 44469321 IC50 > 10000 nM T92609 D0N1HW 5311200 Ki = 2200 nM T92609 D0R2OU 25070031 Ki = 9800 nM T92609 D0U0YR 11520239 Ki = 40 nM T92609 D00OWF 5280953 Ki > 10000 nM T92609 D00KZF 2419 Ki = 130 nM T92609 D01WJZ 60820 Ki = 0.02 nM T92609 D02FNU 56971 Ki = 87 nM T92609 D02LHR 33625 Ki = 3.7 nM T92609 D02ZSU 9838763 EC50 = 158.49 nM T92609 D03QMR 5685 Ki = 0.1585 nM T92609 D04XCQ 10099811 Ki = 0.2 nM T92609 D07BCO 5684 Ki = 18.62 nM T92609 D08OWQ 122295 Ki = 33 nM T92609 D0B1MJ 6918097 Ki = 0.1585 nM T92609 D0B4TT 17747460 Ki = 39.81 nM T92609 D0EE6L 3038495 Ki = 9.15 nM T92609 D0L5TJ 10527469 Ki = 0.22 nM T92609 D0L9SN 4431 Ki = 0.26 nM T92609 D0LL9K 9874983 Ki = 0.36 nM T92609 D0N7LZ 126225 Ki = 25.12 nM T92609 D0P9FT 148842 Ki = 0.34 nM T92609 D0U3HP 164089 Ki = 0.04 nM T92609 D0V8NS 609483 Ki = 1 nM T92609 D0W7IR 9887884 Ki = 1100 nM T92609 D0Z2UD 9872515 Ki = 1 nM T92609 D0Z3UP 216249 EC50 = 25 nM T92609 C9X3BF 4786 EC50 = 230000 nM T92609 C5H9CN 9287 Ki > 10000 nM T92609 C9E6DA 21171 IC50 = 5400 nM T92609 CPK89W 43260 EC50 = 7100 nM T92609 CU86VK 54459 IC50 = 2884.03 nM T92609 C28VFY 60602 Ki = 0.16 nM T92609 CQ3R6M 72457 Ki = 4740 nM T92609 C5Q8JB 76632 EC50 = 11000 nM T92609 CN9GK1 104911 Ki = 20 nM T92609 CT1M8Y 119204 Ki = 251.19 nM T92609 CFD09K 121102 Ki = 2.089 nM T92609 C2H1VA 131829 Ki = 1122.02 nM T92609 CCP43U 146762 EC50 = 25 nM T92609 CY0O6P 151779 Ki = 125.89 nM T92609 CKFG02 172745 Ki > 50000 nM T92609 C3Q2NW 173712 Ki = 150 nM T92609 CVA6M3 179268 Ki = 2140 nM T92609 CZ0D8W 180707 Ki = 26 nM T92609 C28OMN 183528 Ki = 12590 nM T92609 CF4V5Q 185076 Ki = 1479.11 nM T92609 CT6SO0 197001 Ki = 430 nM T92609 CUO7A3 203096 Ki = 158.49 nM T92609 CHLI84 210172 Ki = 42.66 nM T92609 CH6WT3 218362 Ki = 125.89 nM T92609 CQ5Z8Y 294234 Ki = 1995.26 nM T92609 CVE1R0 449646 Ki = 151 nM T92609 C1XTS7 449647 Ki = 13.2 nM T92609 CE8AI0 456386 Ki = 550 nM T92609 C02ZTJ 456387 Ki = 770 nM T92609 C91HBL 541604 Ki = 700 nM T92609 C1TV2F 1070749 Ki > 2700 nM T92609 CZG25W 1376848 Ki = 128 nM T92609 CAQ2J0 3034396 Ki = 1340 nM T92609 CE4KC8 3038603 Ki = 36 nM T92609 C54FEG 3039881 Ki = 12 nM T92609 CS2Q1G 3045401 IC50 = 346.74 nM T92609 C95KAH 3086052 EC50 > 30000 nM T92609 CU4T6Q 3086326 Ki = 5128.61 nM T92609 C8NRQ5 3386873 Ki = 2500 nM T92609 C2ZYB3 3826471 Ki = 31.62 nM T92609 CF6IK7 3894573 Ki = 0.6 nM T92609 CC9V5K 4013695 Ki = 0.2692 nM T92609 CSL05I 5328775 IC50 > 100000 nM T92609 C5K4PX 6603808 Ki = 11.22 nM T92609 C3A1FO 6604789 Ki < 10000 nM T92609 CK1DQ0 6604803 EC50 = 5.623 nM T92609 CZ2M3Q 9794803 EC50 = 17.38 nM T92609 CD47WU 9795167 EC50 = 7.943 nM T92609 CN90IV 9804599 Ki = 1.259 nM T92609 C5Z2KM 9805944 Ki = 9.9 nM T92609 C0L2CT 9808529 Ki = 1.8 nM T92609 CG0I2Z 9816460 EC50 = 4.571 nM T92609 C4TKB3 9816461 EC50 = 50.12 nM T92609 C0HZL7 9816515 EC50 = 3.162 nM T92609 C1XA0W 9816986 EC50 = 31.62 nM T92609 C1X0UA 9817256 EC50 = 12.59 nM T92609 CO9VA3 9820671 IC50 > 1000 nM T92609 C2U3EZ 9822477 Ki = 100 nM T92609 CF0J1A 9822814 Ki = 33.88 nM T92609 C5DB6G 9823115 Ki = 402.56 nM T92609 CMB3R5 9824384 Ki = 0.5888 nM T92609 C6KJ7P 9827677 Ki = 0.2 nM T92609 CQZ6I0 9828476 Ki = 0.2291 nM T92609 C0VO7E 9830292 Ki = 0.37 nM T92609 CHF96B 9837963 EC50 = 10 nM T92609 CCQ9W3 9838192 EC50 = 9 nM T92609 C2EAU0 9838294 EC50 = 63.1 nM T92609 C2O4HM 9838376 EC50 = 4.467 nM T92609 C3XCW9 9840212 EC50 = 79.43 nM T92609 C8TE4O 9844321 Ki = 86.16 nM T92609 CAK7C9 9844511 Ki = 2.1 nM T92609 CXY3Z2 9847196 Ki = 0.868 nM T92609 C5I1XD 9847419 Ki = 8 nM T92609 CQM8A3 9847845 Ki = 2.63 nM T92609 CCB7Z6 9850782 Ki = 1.5 nM T92609 CY2D5T 9851486 Ki = 1.175 nM T92609 C1SEL3 9859855 EC50 = 19.95 nM T92609 CKF2T8 9864325 Ki = 630 nM T92609 CTY02P 9865254 Ki = 4100 nM T92609 C40JBW 9865801 Ki = 0.3981 nM T92609 CAU0X5 9867616 Ki = 8.17 nM T92609 C7WAK9 9872440 Ki = 0.9 nM T92609 CK5BJ6 9872851 Ki = 0.1995 nM T92609 C7ER3F 9881853 EC50 = 2.512 nM T92609 CV2HW7 9883506 Ki = 26.8 nM T92609 C6A9OS 9890459 Ki = 20 nM T92609 C2SN0D 9891166 Ki = 3.1 nM T92609 CD2KC4 9891213 Ki = 0.5012 nM T92609 CQ9WG1 9891937 Ki = 0.7943 nM T92609 CM7H6I 9891967 IC50 = 3.2 nM T92609 CAM25C 9894665 Ki = 0.33 nM T92609 C8HS4Q 9895326 Ki = 1.072 nM T92609 C5Y2AZ 9895338 Ki = 0.6607 nM T92609 CK7C9L 9903313 EC50 = 50.12 nM T92609 C8RZ7N 9903932 EC50 = 6.31 nM T92609 CFI97S 9904205 IC50 = 537.03 nM T92609 CYWQ50 9906447 Ki > 10000 nM T92609 C7JFZ5 9906978 Ki = 34 nM T92609 CY2I0L 9908478 Ki = 1000 nM T92609 C7SMT0 9908904 IC50 > 1000 nM T92609 CI1H6U 9909211 Ki = 2 nM T92609 CA0U4Y 9909471 Ki = 54.61 nM T92609 C0Y4CZ 9913449 Ki = 0.077 nM T92609 C5THY1 9913616 IC50 = 1.9 nM T92609 CBX74I 9915831 Ki = 1.5 nM T92609 CT6QX7 9916549 Ki = 0.19 nM T92609 C7SOT8 9929936 Ki = 95.42 nM T92609 C1C5KY 9931327 Ki = 4400 nM T92609 C4L1GA 9934033 IC50 = 300 nM T92609 C06OWM 9934955 Ki = 1700 nM T92609 CY8XG3 9938248 Ki = 140 nM T92609 CUQ8I5 9947861 EC50 = 2.818 nM T92609 CO2X8D 9951544 IC50 = 213.8 nM T92609 C4G9VQ 9954092 Ki = 130 nM T92609 CD97EL 9959671 Ki = 0.1 nM T92609 C6LZS7 9959689 Ki = 0.4 nM T92609 CW89JP 9960311 Ki = 3.05 nM T92609 CF1C5Q 9960497 Ki = 0.32 nM T92609 C7JXL1 9976756 Ki = 37.15 nM T92609 C2WVQ9 9982050 Ki = 1.1 nM T92609 CF7QK6 9982585 Ki = 1.3 nM T92609 C6PCS8 9984150 Ki = 1.7 nM T92609 CD0IS5 9985476 Ki = 0.12 nM T92609 C4IG8L 10005161 Ki = 0.19 nM T92609 CA29FW 10015132 EC50 = 12.59 nM T92609 C6XGV2 10020855 Ki = 33 nM T92609 CRH7V9 10026936 Ki = 2 nM T92609 CGN05I 10029146 Ki = 0.51 nM T92609 C05ICW 10031709 Ki = 0.1 nM T92609 CZX09T 10038958 EC50 = 12.59 nM T92609 C3A1ME 10047430 Ki = 0.9 nM T92609 C9P4AC 10048729 Ki = 1.93 nM T92609 C71CVU 10060965 EC50 = 3.162 nM T92609 C0I2RV 10065903 Ki = 954.99 nM T92609 CDF0Z2 10071710 Ki = 3.311 nM T92609 CCN5S8 10073934 IC50 = 1910 nM T92609 CN9B1F 10074286 Ki = 0.18 nM T92609 CVD98U 10083742 EC50 = 39.81 nM T92609 CKA5F4 10084076 Ki = 373 nM T92609 CSW74O 10084685 EC50 = 25.12 nM T92609 CC2ZY0 10089254 Ki = 15.85 nM T92609 C0IWD7 10091187 Ki = 4.98 nM T92609 C8NQ3I 10092649 Ki = 11 nM T92609 C3SJX0 10095044 Ki = 1.4 nM T92609 CP51OC 10097317 Ki = 2 nM T92609 CLW53J 10097792 Ki = 0.3236 nM T92609 CA5H7K 10106205 Ki = 200 nM T92609 C54EYD 10108561 IC50 = 398.11 nM T92609 CE27RV 10135864 EC50 = 219 nM T92609 COPD43 10160408 IC50 = 1.9 nM T92609 C2B5SJ 10180440 EC50 = 252 nM T92609 CUN52S 10183297 Ki = 200 nM T92609 CSJ40T 10198532 EC50 = 2.512 nM T92609 CJ31LA 10199052 EC50 = 15.85 nM T92609 C7MKP9 10199335 EC50 = 16.6 nM T92609 CU2B9P 10221004 EC50 = 239.88 nM T92609 CX9YD5 10221005 EC50 = 1.95 nM T92609 C12UXA 10221066 EC50 = 25.12 nM T92609 CO64WJ 10236758 Ki = 436.52 nM T92609 CCF6U9 10244367 EC50 = 3.311 nM T92609 CVF1E5 10246054 IC50 = 162.18 nM T92609 C8SYA1 10252540 Ki = 12.3 nM T92609 CBCZ21 10256583 Ki = 1.59 nM T92609 C9KDO8 10287924 Ki = 314 nM T92609 C0U3WR 10314056 Ki = 793 nM T92609 C62PAC 10318686 Ki = 1.1 nM T92609 C3E5CB 10337773 Ki = 25118.86 nM T92609 C06YPQ 10342554 Ki = 1.2 nM T92609 CIP38T 10344976 Ki = 0.4169 nM T92609 C3YB4P 10345121 IC50 = 1920 nM T92609 CSB63G 10345845 IC50 > 10000 nM T92609 CI17PT 10348924 Ki = 0.73 nM T92609 C7P8RU 10357155 IC50 > 100000 nM T92609 C5HQ2A 10362296 Ki = 100 nM T92609 COC7M0 10363912 Ki = 19.5 nM T92609 C0W8QR 10364538 Ki > 2000 nM T92609 C8GR5I 10364994 Ki = 0.4677 nM T92609 CS7F3J 10371061 Ki = 0.2 nM T92609 CE9IN1 10378649 EC50 = 19.95 nM T92609 C4H6YF 10379435 EC50 = 56.23 nM T92609 CDAC63 10381889 IC50 = 14.45 nM T92609 C3N7TF 10382537 Ki = 977.24 nM T92609 C7W4TF 10391177 IC50 = 1000 nM T92609 CSAF82 10393665 Ki = 0.4 nM T92609 CG1IR6 10394346 Ki = 1.8 nM T92609 C0MBY3 10399043 EC50 = 51.29 nM T92609 CS6MA7 10413283 IC50 = 600 nM T92609 CQ52MH 10414908 Ki = 0.48 nM T92609 C7Z5FO 10415038 Ki = 0.69 nM T92609 C9EIT6 10415156 Ki = 0.7 nM T92609 C7LGR3 10420352 EC50 = 3300 nM T92609 CM76FU 10422033 EC50 = 20.89 nM T92609 C0R3LA 10423384 EC50 = 25.12 nM T92609 CP7B3M 10430193 Ki = 9.12 nM T92609 CCP0S9 10434440 Ki = 0.63 nM T92609 CIQ02H 10436842 Ki = 0.8 nM T92609 CZTU54 10437624 Ki = 0.6 nM T92609 CQ93PA 10438280 Ki = 0.1 nM T92609 C58HNW 10473406 Ki = 7300 nM T92609 C7GEB0 10474042 Ki = 0.33 nM T92609 C0D1VZ 10479323 Ki = 85.11 nM T92609 CW16TJ 10481087 Ki = 0.99 nM T92609 C6UFO7 10506484 Ki = 1 nM T92609 C85BUY 10506673 Ki = 0.9 nM T92609 CX73IB 10506729 Ki = 0.41 nM T92609 CY84UO 10507089 Ki = 1.02 nM T92609 C69OVN 10507129 Ki = 8 nM T92609 CMG18U 10507220 Ki = 0.5 nM T92609 C3KX6O 10507357 Ki = 6.9 nM T92609 C6C1NB 10507411 Ki = 1.1 nM T92609 CKJI08 10507500 Ki = 0.2 nM T92609 CJ0K1T 10507651 Ki = 8.913 nM T92609 C2U8AC 10508016 Ki = 36.31 nM T92609 C4XZ3Y 10508132 Ki = 58.88 nM T92609 C0U9GR 10508330 Ki = 0.2 nM T92609 CZP09X 10508332 Ki = 1.479 nM T92609 CR0XV8 10530491 Ki = 0.16 nM T92609 C35RPS 10530552 Ki = 0.6 nM T92609 C41XOR 10531022 Ki = 1.5 nM T92609 C0D4VW 10531157 Ki = 0.01 nM T92609 CE82ZX 10531476 Ki = 0.1 nM T92609 C4X9EF 10531532 Ki = 8.71 nM T92609 CJ3CL2 10531675 Ki = 1.9 nM T92609 C7MI2N 10531766 Ki = 1.122 nM T92609 CCQI21 10532044 Ki = 4.786 nM T92609 C8PA4X 10549596 Ki = 0.912 nM T92609 CH8W9A 10554140 Ki = 0.2 nM T92609 CCKT30 10554745 Ki = 4.2 nM T92609 CPE27N 10554913 Ki = 0.7 nM T92609 C8NXE5 10554957 Ki = 0.4 nM T92609 C2ONS3 10555024 Ki = 0.2 nM T92609 CV7F9T 10555223 Ki = 10 nM T92609 C16APC 10555288 Ki = 1.1 nM T92609 CQ29UC 10555618 Ki = 3.715 nM T92609 C7ROD9 10556164 Ki = 0.4 nM T92609 C2WGC8 10575494 Ki = 19.38 nM T92609 CQXU07 10575664 Ki = 18.95 nM T92609 CY04PF 10577609 Ki = 1112.8 nM T92609 C7LWD8 10578548 Ki = 1.2 nM T92609 C93CLB 10578715 Ki = 0.11 nM T92609 C18HKX 10578735 Ki = 14 nM T92609 CT0ML5 10578926 Ki = 20 nM T92609 C4SVP1 10578990 Ki = 1.47 nM T92609 CF24MW 10579368 Ki = 316.23 nM T92609 C2LRK3 10579632 Ki = 5 nM T92609 CFQB52 10580182 Ki = 1.7 nM T92609 CWM6C3 10599007 Ki = 0.35 nM T92609 CZ8IX1 10602912 Ki = 0.46 nM T92609 CR8ZX2 10603727 Ki = 1.2 nM T92609 CD7W1O 10603739 Ki = 0.8 nM T92609 CK8SO7 10603951 Ki = 20.42 nM T92609 C72ELH 10615770 IC50 > 100000 nM T92609 C8YXF5 10616819 IC50 > 100000 nM T92609 C2G4IR 10617200 Ki = 36.31 nM T92609 C8B5CJ 10621590 Ki = 16.6 nM T92609 CE5CU8 10621592 Ki = 23.99 nM T92609 CC34GW 10626453 Ki = 22 nM T92609 CY4H5J 10626493 Ki = 0.3 nM T92609 COU08R 10626610 Ki = 1 nM T92609 C6BHD5 10626686 Ki = 8 nM T92609 CNE1X0 10626726 Ki = 0.2 nM T92609 CUF48J 10626772 Ki = 0.4 nM T92609 CVG42P 10626843 Ki = 0.5 nM T92609 CQ13HM 10626910 Ki = 0.23 nM T92609 CXD31C 10626911 Ki = 0.77 nM T92609 CB26QH 10626982 Ki = 56.23 nM T92609 CYG6R7 10627003 Ki = 0.76 nM T92609 CSWC40 10627021 Ki = 1.38 nM T92609 CFA2R6 10627090 Ki = 0.1 nM T92609 C3TSO7 10627094 Ki = 1.6 nM T92609 CDC19N 10627155 Ki = 0.2 nM T92609 CF38IK 10627279 Ki = 2.1 nM T92609 CZ3T7S 10627329 Ki = 4.9 nM T92609 CER8L0 10640982 Ki = 389.05 nM T92609 C70QNW 10649481 Ki = 0.14 nM T92609 C9VY7F 10650129 Ki = 0.4 nM T92609 C6J4OK 10650633 Ki = 1.2 nM T92609 C4HP6A 10650726 Ki = 0.1 nM T92609 CLV1Q4 10650843 Ki = 0.95 nM T92609 CF1P6Z 10651080 Ki = 8.71 nM T92609 CBN78H 10651219 Ki = 0.1 nM T92609 CV2HA5 10651636 Ki = 0.06 nM T92609 C3K7UP 10651654 Ki = 1.862 nM T92609 C07UGY 10673657 Ki = 0.12 nM T92609 CG6P7N 10674055 Ki = 0.2 nM T92609 C35NWA 10674133 Ki = 4.25 nM T92609 CRQD91 10674333 Ki = 0.7 nM T92609 CX69JL 10674544 Ki = 4.5 nM T92609 CQ9JN3 10674564 Ki = 0.18 nM T92609 C4EC8H 10674791 Ki = 4.5 nM T92609 C95VPX 10674840 Ki = 0.8 nM T92609 CTB7L2 10674896 Ki = 1.82 nM T92609 CC8IT7 10675068 Ki = 0.2 nM T92609 CBEP65 10688604 Ki = 77.62 nM T92609 CB0F2I 10697623 Ki = 0.18 nM T92609 CA80KS 10697912 Ki = 0.6 nM T92609 C16NJO 10698141 Ki = 0.8 nM T92609 C6PVI9 10698570 Ki = 0.05 nM T92609 C4XZM6 10698974 Ki = 19 nM T92609 CI4V5M 10699164 Ki = 0.08 nM T92609 C0HO7D 10720893 Ki = 0.2 nM T92609 C87QBC 10721171 Ki = 0.3 nM T92609 C5WR2P 10721476 Ki = 0.3 nM T92609 C3WQ9B 10721564 Ki = 0.75 nM T92609 CZI63U 10721568 Ki = 0.88 nM T92609 C5L4AS 10721730 Ki = 7.9 nM T92609 CPF96G 10722045 Ki = 0.2 nM T92609 C6N7CQ 10722099 Ki = 0.3 nM T92609 CE2GK7 10739024 Ki = 830 nM T92609 C1QZ3O 10743042 Ki = 5.93 nM T92609 CGQ8I3 10744391 Ki = 11 nM T92609 CU6HM4 10745305 Ki = 3.6 nM T92609 CHT1L0 10745380 Ki = 0.1 nM T92609 C1RZU6 10745566 Ki = 14 nM T92609 CA17HU 10745664 Ki = 12 nM T92609 CW91BJ 10745766 Ki = 0.7 nM T92609 C6IG0M 10745901 Ki = 0.02 nM T92609 CS3ON2 10746137 Ki = 5.2 nM T92609 CJ8VM0 10747021 Ki = 6.9 nM T92609 CBZP19 10747201 Ki = 0.1 nM T92609 C51YSW 10764133 Ki = 812.83 nM T92609 CFM65K 10767981 Ki = 1.862 nM T92609 C0WMG4 10768610 Ki = 22 nM T92609 C58CRB 10768829 Ki = 0.3 nM T92609 CV1JT2 10769037 Ki = 3.2 nM T92609 C63FIL 10769058 Ki = 1.1 nM T92609 CT1K3B 10769331 Ki = 0.5248 nM T92609 C6JG4Z 10769621 Ki = 0.3 nM T92609 CV6T3C 10770007 Ki = 0.3 nM T92609 C8LZM3 10770057 Ki = 1.19 nM T92609 C9ARF0 10770317 Ki = 1.22 nM T92609 CS8QR2 10787126 Ki = 18.2 nM T92609 C87POR 10790430 Ki = 8.7 nM T92609 C1RC8F 10790988 Ki = 23.72 nM T92609 CMU59N 10791843 Ki = 2.3 nM T92609 C4XK8Y 10792591 Ki = 2.2 nM T92609 CS24OF 10792897 Ki = 0.29 nM T92609 C6F5HP 10792898 Ki = 0.66 nM T92609 CN71ZB 10793023 Ki = 1.8 nM T92609 C3O7YN 10793665 Ki = 1.778 nM T92609 CTXB06 10793720 Ki = 0.98 nM T92609 C0D6MW 10793963 Ki = 5.888 nM T92609 C5W7FC 10804826 EC50 = 24547.09 nM T92609 C6EWQ3 10811627 Ki = 8.4 nM T92609 CXU6D7 10815549 Ki = 0.4 nM T92609 CN6ZP7 10815593 Ki = 0.12 nM T92609 C4ZNR1 10816815 Ki = 0.4 nM T92609 C68UVF 10816832 Ki = 3.5 nM T92609 CO73GU 10816903 Ki = 16 nM T92609 CID39T 10817365 Ki = 0.06 nM T92609 CO23UP 10817661 Ki = 3.631 nM T92609 CBO8N9 10818003 Ki = 53.7 nM T92609 CFC95U 10834793 Ki = 0.6457 nM T92609 C5NFU1 10836245 Ki = 0.3 nM T92609 CIY58E 10839105 Ki = 0.18 nM T92609 CKS74R 10839106 Ki = 20 nM T92609 C5SC1X 10839825 Ki = 0.39 nM T92609 CP78AK 10840177 Ki = 0.5 nM T92609 C49YSD 10840781 Ki = 430 nM T92609 C4LV0H 10841070 Ki = 0.33 nM T92609 CE80NV 10841190 Ki = 7.079 nM T92609 C2RXD0 10841296 Ki = 6.8 nM T92609 CYSL64 10841387 Ki = 3.1 nM T92609 C8TED5 10841819 Ki = 7.5 nM T92609 CO9WP2 10841851 Ki = 1.3 nM T92609 C70LSM 10880840 Ki > 1000 nM T92609 C3I1CT 10892762 Ki = 201 nM T92609 CEUD36 10893672 Ki = 18.56 nM T92609 C8VT6G 10916464 Ki = 457.09 nM T92609 CBH30I 10916771 Ki = 0.22 nM T92609 CD7QW2 10917316 Ki = 0.53 nM T92609 CH95TI 10923927 Ki = 616.6 nM T92609 C0N6KJ 10928520 Ki = 1 nM T92609 C3CI6Z 10934575 EC50 = 0.1096 nM T92609 C8LPD2 10939209 Ki = 26 nM T92609 C69ULE 10939408 Ki = 104 nM T92609 CTO4Z9 10949698 Ki = 0.89 nM T92609 CAIJ61 10961351 Ki = 0.32 nM T92609 CP5KV2 10962489 Ki = 24.54 nM T92609 CW6T1N 10971791 Ki = 3.02 nM T92609 CX5M6J 10974101 Ki = 0.16 nM T92609 CUK3X0 10982853 Ki = 48 nM T92609 CC2NG9 10994812 Ki = 0.44 nM T92609 C2BF0W 11014848 Ki = 2.29 nM T92609 CGW87Y 11034737 EC50 = 10.47 nM T92609 CZM27Y 11039289 Ki = 0.094 nM T92609 CH9O0P 11046644 Ki = 1.62 nM T92609 CD0H8T 11049096 Ki = 33.88 nM T92609 C48QYR 11058166 EC50 = 41.69 nM T92609 C7JI1M 11059195 EC50 = 1096.48 nM T92609 C7R2AZ 11079593 EC50 = 436.52 nM T92609 CUZ38C 11081136 Ki = 2 nM T92609 C91BKL 11090351 EC50 = 23.99 nM T92609 CF32NC 11092254 Ki = 0.28 nM T92609 CFE1M7 11097789 EC50 = 7.762 nM T92609 CTG4I5 11098175 EC50 = 1.585 nM T92609 C84VUJ 11108001 EC50 = 5.012 nM T92609 CR6K4V 11109088 EC50 = 0.4365 nM T92609 CJT65Y 11123606 Ki = 1.51 nM T92609 CF68CS 11133288 Ki = 0.3981 nM T92609 C7MD3R 11133868 Ki = 2.344 nM T92609 C3ZJK1 11134424 Ki = 0.3 nM T92609 CC0HY8 11135150 Ki = 100 nM T92609 CG40BP 11140345 EC50 = 7.762 nM T92609 CO0XW1 11140347 EC50 = 2.291 nM T92609 CA7Y5Z 11144555 Ki = 2.59 nM T92609 C73DFT 11145007 Ki = 2.99 nM T92609 CUNH28 11152823 Ki = 158.49 nM T92609 C0W4OI 11154198 Ki = 2.818 nM T92609 C7VKQ5 11164948 Ki = 2570.4 nM T92609 CUE3X2 11176459 Ki = 169.82 nM T92609 CSFD06 11189150 Ki = 1.4 nM T92609 CQ9NP6 11198145 IC50 = 100 nM T92609 C4J8YG 11211017 Ki = 620 nM T92609 CR10CS 11234230 Ki = 70.04 nM T92609 CP9U5C 11264016 EC50 = 30000 nM T92609 CKEJ43 11270912 Ki = 1.445 nM T92609 C90UKI 11281005 Ki = 25.12 nM T92609 CR2DJ1 11282574 Ki = 288.4 nM T92609 C1VNU0 11303180 Ki = 23.4 nM T92609 CCQ0S5 11338016 Ki = 95.5 nM T92609 CT3V5I 11338314 Ki = 3800 nM T92609 CTB03C 11372228 Ki = 43.14 nM T92609 C4SZ7W 11384664 Ki = 29.9 nM T92609 C7KX6F 11430126 Ki = 0.8128 nM T92609 C7EVT0 11430491 Ki = 0.2884 nM T92609 CM8I7N 11454386 Ki = 1.413 nM T92609 C89FRU 11464777 Ki = 149.34 nM T92609 C8Q1LZ 11486511 Ki = 234.42 nM T92609 C8TDA7 11488170 Ki = 977.24 nM T92609 COI68V 11496213 Ki = 21 nM T92609 CI62OX 11502343 IC50 = 1800 nM T92609 CPO8S1 11502381 IC50 = 4500 nM T92609 C2TVA0 11502638 IC50 = 5900 nM T92609 CTMH12 11505007 Ki = 1.2 nM T92609 CF45XR 11511026 Ki = 46 nM T92609 CS24AX 11516386 IC50 = 2900 nM T92609 C20FMG 11517340 IC50 > 10000 nM T92609 CPQN50 11517341 IC50 = 4200 nM T92609 CS20NG 11519153 Ki = 0.91 nM T92609 CL09JW 11524225 IC50 = 10000 nM T92609 CI8GN0 11532563 Ki = 1.99 nM T92609 C8GZ1I 11539020 IC50 > 10000 nM T92609 C0MF3O 11539392 Ki = 1.585 nM T92609 C0ZBJ6 11554490 Ki = 68 nM T92609 COC6U3 11554541 Ki = 1.259 nM T92609 CZMB92 11567596 IC50 = 6200 nM T92609 CEV2P7 11567620 Ki = 9 nM T92609 CP7W6H 11567952 IC50 > 10000 nM T92609 CR7M5S 11568725 Ki = 58 nM T92609 CE0U8J 11581337 IC50 = 2200 nM T92609 C2IE4D 11583392 Ki = 0.2512 nM T92609 CS1OR8 11584530 Ki = 119 nM T92609 C6D1MA 11584660 Ki > 630.96 nM T92609 C1M2CP 11589069 Ki = 42 nM T92609 C3V6LN 11590801 Ki = 12 nM T92609 CJW9E6 11604548 Ki = 1.99 nM T92609 CD28IH 11618024 IC50 = 6300 nM T92609 C36OSA 11618702 IC50 = 6500 nM T92609 C6JRN0 11619713 Ki = 7.943 nM T92609 C3IHP8 11626704 Ki = 0.251 nM T92609 C9VAI5 11633517 Ki = 0.3981 nM T92609 C5W0JR 11633992 Ki = 72 nM T92609 CL6XP8 11638677 Ki = 3.467 nM T92609 CI2KZ1 11641036 IC50 = 7200 nM T92609 CZA0M9 11653915 Ki = 19.9 nM T92609 CJV2I4 11655403 Ki = 227 nM T92609 CX7FR8 11655728 Ki = 2.754 nM T92609 C6URZ0 11668565 Ki = 10 nM T92609 CJSN27 11668594 IC50 = 1100 nM T92609 C9I7KB 11669646 Ki = 1.995 nM T92609 C87TCD 11689687 IC50 = 1300 nM T92609 CUVL17 11705133 Ki = 1.995 nM T92609 C2E8BF 11705395 Ki = 60 nM T92609 CL08TQ 11711943 Ki = 272 nM T92609 C7RAS6 11712250 Ki = 1.413 nM T92609 C7PK3H 11712470 Ki = 0.316 nM T92609 CR1L6N 11732516 Ki = 162.8 nM T92609 C12YTV 11742585 Ki = 1670 nM T92609 CJ60OP 11742834 Ki = 0.05012 nM T92609 C3G4FS 11751173 Ki = 1.259 nM T92609 CO50RT 11757736 Ki = 0.5 nM T92609 C06HZD 11782656 Ki = 14.6 nM T92609 C28UNM 11784634 Ki = 1698.24 nM T92609 C4VL6W 11801214 Ki = 2.09 nM T92609 C87FWQ 11801562 Ki = 3.548 nM T92609 CFTI34 11801828 Ki = 16.22 nM T92609 C4ZXG0 11801861 Ki = 81 nM T92609 C2RPQ0 11802456 Ki = 0.1 nM T92609 C1VWL5 11811395 EC50 = 1949.84 nM T92609 CUB53N 11857638 Ki = 1.8 nM T92609 C29HBR 11857639 Ki = 1.4 nM T92609 C29FMG 11857709 Ki = 1.8 nM T92609 CX50UR 11857710 Ki = 1.3 nM T92609 CW6V5E 11857711 Ki = 1.8 nM T92609 CD50HW 11857791 Ki = 2.2 nM T92609 CGL5D9 11857792 Ki = 6.2 nM T92609 CE0U9G 11857793 Ki = 4.8 nM T92609 CYJ5I7 11857794 Ki = 7 nM T92609 C9S5NU 11857861 Ki = 8.5 nM T92609 CU83FA 11857862 Ki = 12 nM T92609 CUO32E 11857863 Ki = 16 nM T92609 CD7O6J 11857864 Ki = 3.3 nM T92609 CXLW54 11948707 Ki = 413 nM T92609 C8JQL7 11957735 IC50 > 10000 nM T92609 CH1WZ3 11984570 Ki = 0.2 nM T92609 CJP2T4 11994550 Ki = 11.48 nM T92609 CHE4O6 11994665 Ki = 1.202 nM T92609 C0ZRF5 11994667 Ki = 5.623 nM T92609 CQW63S 11994668 Ki = 16.22 nM T92609 CVNL73 11994670 Ki = 234.42 nM T92609 C1BZQ0 11994673 Ki = 66.07 nM T92609 CB3DJ5 11994797 Ki = 2.818 nM T92609 C1KQO2 11994915 Ki = 87.1 nM T92609 CU17YO 11995033 Ki = 9.333 nM T92609 C3F1BT 11995035 Ki = 323.59 nM T92609 C1A2IB 12001199 Ki < 1995.26 nM T92609 C8W5JG 12039032 Ki = 417 nM T92609 CY8DS2 12134985 Ki = 79 nM T92609 C4CI5P 12134986 Ki = 3.8 nM T92609 CS6BU1 12134987 Ki = 89 nM T92609 CPX75G 12134991 Ki = 2321 nM T92609 CI52SU 12134994 Ki = 578 nM T92609 C8WEX1 12134995 Ki = 202 nM T92609 C6S9BY 12134996 Ki = 40 nM T92609 C2U3RT 12764879 EC50 = 70 nM T92609 C0B1QO 12764880 EC50 = 721 nM T92609 CFN31J 12840734 Ki = 2684 nM T92609 C8H4TF 12924821 EC50 = 120 nM T92609 C2V9FL 13091268 Ki = 39.3 nM T92609 CMA46J 13305910 Ki = 0.4074 nM T92609 CN2ZQ5 13911290 Ki = 0.344 nM T92609 CV08GM 14378574 Ki = 616 nM T92609 C4E7NH 14423371 Ki = 0.166 nM T92609 CMO81H 14925759 Ki = 53.7 nM T92609 C8BF2P 15254720 Ki = 25.12 nM T92609 CQ5ZJ2 15546405 Ki = 53 nM T92609 C1CX2S 15675860 Ki < 100000 nM T92609 CRTO23 15840661 Ki = 1 nM T92609 CPR25X 15986917 Ki < 2511.89 nM T92609 C5KW3L 15987108 Ki < 1995.26 nM T92609 CXW37K 15987265 IC50 = 3200 nM T92609 CT03WI 16040907 Ki = 38 nM T92609 CW5NS1 16041090 Ki = 74 nM T92609 C03VCW 16041091 Ki = 11 nM T92609 CM3O4Z 16041092 Ki = 3.6 nM T92609 CUL5M9 16041263 Ki = 11 nM T92609 C6S8AM 16041264 Ki = 5.1 nM T92609 CYTD80 16041265 Ki = 6.2 nM T92609 C86MYV 16041449 Ki = 6.5 nM T92609 CHF7K6 16041451 Ki = 34 nM T92609 CCJ65Y 16041628 Ki = 3.1 nM T92609 CE2Z7Y 16041629 Ki = 1.7 nM T92609 CRJX49 16041630 Ki = 5.3 nM T92609 CDTN28 16121006 Ki = 1.585 nM T92609 C6NRI4 16219720 Ki = 0.16 nM T92609 CERP08 16219807 Ki < 10000 nM T92609 CI8DR5 16638286 IC50 = 462 nM T92609 CZ2IS9 16660294 Ki > 10000 nM T92609 CZ8S6B 16721032 Ki = 23.44 nM T92609 C7KS8E 16721110 Ki = 1.318 nM T92609 C4NC3P 16756752 Ki = 34000 nM T92609 CWF10J 16756753 Ki = 1010 nM T92609 C3GD2P 17753379 Ki = 1 nM T92609 CM60NI 17804479 EC50 = 385 nM T92609 CN0CH5 18187410 Ki = 0.28 nM T92609 CT3OK4 18738380 Ki = 28 nM T92609 CF1DM9 18738384 Ki = 1.8 nM T92609 CEP14V 18738385 Ki = 0.5 nM T92609 CM6YI0 18738386 Ki = 0.2 nM T92609 CCO79B 18738387 Ki = 14 nM T92609 C9E4ID 18738412 Ki = 1502 nM T92609 CYT58A 19085820 Ki = 0.13 nM T92609 CHM64Z 19085827 Ki = 499 nM T92609 CV8X0D 19085829 Ki = 0.27 nM T92609 C9CL0I 19085832 Ki = 20 nM T92609 C2EYW8 19085836 Ki = 147 nM T92609 C6KSV0 19085839 Ki = 3.1 nM T92609 CRU75T 19085858 Ki = 0.057 nM T92609 CN5XJ1 19085866 Ki = 0.12 nM T92609 C2L1IX 19085869 Ki = 1.2 nM T92609 C4V1LT 19085876 Ki = 0.084 nM T92609 C7A2EC 19085881 Ki = 0.16 nM T92609 C8RDC1 19085894 Ki = 2.4 nM T92609 CC1Y7N 19085914 Ki = 0.064 nM T92609 C7T6HA 19085921 Ki = 1033 nM T92609 C7M9NZ 19085926 Ki = 0.099 nM T92609 C6AOE8 19426635 IC50 = 190.55 nM T92609 CRF1H4 19608536 Ki = 50.2 nM T92609 CPJG69 20215436 Ki = 1.39 nM T92609 C4GM9S 20750645 Ki = 331 nM T92609 CPRJ25 21392988 Ki = 107151.93 nM T92609 C3T5HF 21509921 Ki = 2371 nM T92609 CD9Y0E 21712258 Ki = 7.3 nM T92609 CEI9P4 21823379 IC50 = 552.3 nM T92609 CT7XG9 21830793 Ki = 6.75 nM T92609 C8GUJ3 22120322 IC50 = 288.4 nM T92609 CGO3B8 22120332 IC50 = 114.82 nM T92609 C21LHM 22493224 EC50 = 12.59 nM T92609 C4UYD5 22493225 EC50 = 1000 nM T92609 C9V4MO 22493231 EC50 = 398.11 nM T92609 CKB2N6 22493233 EC50 = 50.12 nM T92609 C0P2UY 22493236 EC50 = 0.7943 nM T92609 C02AEX 22493245 Ki = 2187.76 nM T92609 CWT85U 22493254 EC50 = 87.1 nM T92609 CK8GD3 22493257 EC50 = 125.89 nM T92609 C09UWJ 22493258 EC50 = 1 nM T92609 C6BTO5 22493263 EC50 = 1.259 nM T92609 C7NGV2 22493265 EC50 = 12.59 nM T92609 CJ1G5C 22493269 EC50 = 15.14 nM T92609 CR63XU 22493272 EC50 = 323.59 nM T92609 CGI40S 22493274 EC50 = 12.59 nM T92609 C3JW1Q 22493280 EC50 = 0.7943 nM T92609 CG28DA 22493287 EC50 = 676.08 nM T92609 CYHG72 22493289 EC50 = 10 nM T92609 CMS13N 22493316 EC50 < 100000 nM T92609 C6ADV8 22493318 EC50 = 0.4677 nM T92609 CS4EI0 22493320 EC50 = 19.95 nM T92609 CSF43L 22493325 EC50 = 660.69 nM T92609 C1QOL5 22493343 EC50 = 1.995 nM T92609 CKIJ24 22493344 EC50 = 316.23 nM T92609 C7FCZ5 22493347 EC50 = 52.48 nM T92609 CDE4R9 22493349 EC50 = 38.9 nM T92609 CSCP16 22493352 EC50 = 0.6607 nM T92609 C3N9RK 22493356 EC50 = 24.55 nM T92609 C7XEF1 22493359 EC50 = 724.44 nM T92609 C5ZNB0 22493365 EC50 = 1.259 nM T92609 CI1GH6 22493367 EC50 = 199.53 nM T92609 C86PSG 22493372 EC50 = 109.65 nM T92609 CI42EA 22493379 EC50 = 50.12 nM T92609 CY80ON 22493381 EC50 = 398.11 nM T92609 C4LJO9 22493387 EC50 < 100000 nM T92609 CP34UB 22493392 EC50 = 6.761 nM T92609 C9DS1F 22493401 EC50 = 100 nM T92609 CAFG09 22493408 EC50 = 794.33 nM T92609 C9T5VN 22493411 EC50 = 501.19 nM T92609 CM86HE 22493415 EC50 = 42.66 nM T92609 C81XUE 23027035 IC50 > 10000 nM T92609 CR5H1I 23027211 IC50 > 10000 nM T92609 CC2L1B 23027245 IC50 = 3000 nM T92609 CG9M4Y 23027411 IC50 > 10000 nM T92609 CC6R2O 23027527 IC50 = 7500 nM T92609 C6QC2D 23151199 IC50 = 6500 nM T92609 C0NI3J 23290944 Ki = 584 nM T92609 CL1YH7 23582308 Ki = 50.12 nM T92609 CRN13C 24748804 Ki < 2511.89 nM T92609 C96KDH 24748992 Ki < 1584.89 nM T92609 CH8N1W 24748993 Ki < 1995.26 nM T92609 CRGJ52 24749183 Ki < 3981.07 nM T92609 C13GRZ 24749184 Ki < 3981.07 nM T92609 C8ZE6H 24749185 Ki < 3162.28 nM T92609 CWTB59 24749606 Ki < 2511.89 nM T92609 CT93NP 24749721 Ki < 3981.07 nM T92609 CI6W7D 24749841 Ki < 10000 nM T92609 C20QND 24749960 Ki < 3981.07 nM T92609 CSXA65 24749962 Ki < 1995.26 nM T92609 CUX7C3 24803316 Ki = 316.23 nM T92609 C1QTN4 24803480 Ki = 1584.89 nM T92609 CTU67D 24803482 Ki = 31.62 nM T92609 C31QHW 24803483 Ki = 25.12 nM T92609 C3RYC2 24803638 Ki = 63.1 nM T92609 CI4EA6 24803639 Ki = 100 nM T92609 CJ07ES 24803641 Ki = 100 nM T92609 C04KHJ 24803797 Ki = 31.62 nM T92609 CY26TH 24803798 Ki = 125.89 nM T92609 C50BOH 24803799 Ki = 158.49 nM T92609 C2AKX9 24804150 Ki = 31.62 nM T92609 C9K0CX 24805674 Ki = 6 nM T92609 C58AMS 24829343 Ki = 71.3 nM T92609 CDC91N 24839550 Ki = 1659.59 nM T92609 CUW23K 24854106 Ki = 20 nM T92609 CX6R0P 24894141 Ki = 165.96 nM T92609 C5QG6V 24894147 Ki = 3.388 nM T92609 CW2FG9 24897950 Ki = 0.6026 nM T92609 C1VRJ3 25014630 IC50 = 1900 nM T92609 CKR94M 25022356 Ki = 100 nM T92609 CA20NZ 25025581 Ki = 199.53 nM T92609 CMVL70 25059766 IC50 > 1000 nM T92609 CED30A 25059770 IC50 > 1000 nM T92609 CJU9Y7 25060021 IC50 > 1000 nM T92609 C36PMH 25060023 IC50 > 1000 nM T92609 CHSB87 25060024 IC50 > 1000 nM T92609 CJOY17 25066019 EC50 = 43 nM T92609 COE3T5 25071310 Ki = 1258.93 nM T92609 CZ48AL 25071621 Ki = 199.53 nM T92609 C6I7JN 25071929 Ki = 39.81 nM T92609 CFE62W 25071930 Ki = 100 nM T92609 CU0SR4 25071931 Ki = 1995.26 nM T92609 C18XGM 25072242 Ki = 100 nM T92609 C4RE0M 25072246 Ki > 2511.89 nM T92609 CTWZ82 25072568 Ki > 2511.89 nM T92609 CW2H9F 25072875 Ki = 1584.89 nM T92609 CA4FV9 25072876 Ki = 1258.93 nM T92609 CPUB18 25072877 Ki > 2511.89 nM T92609 C6GPL3 25072880 Ki = 794.33 nM T92609 CDY9Z4 25073188 Ki > 2511.89 nM T92609 C3AJD0 25073189 Ki = 794.33 nM T92609 C9KR8V 25073190 Ki > 2511.89 nM T92609 C68FHZ 25073191 Ki = 1995.26 nM T92609 C98ISN 25073801 Ki = 501.19 nM T92609 CF7P2A 25130875 Ki = 158.49 nM T92609 C7P1QS 25130876 Ki = 436.52 nM T92609 C6G5BO 25130877 Ki > 1000 nM T92609 CL8GD3 25130878 Ki > 1000 nM T92609 CT78MG 25130879 Ki = 199.53 nM T92609 C7WXA2 25131192 Ki = 467.74 nM T92609 C3UVA0 25131193 Ki = 338.84 nM T92609 C0GM3L 25131196 Ki = 537.03 nM T92609 CFUT35 25131198 Ki = 169.82 nM T92609 C1Y3TS 25131871 Ki > 1000 nM T92609 CFJ6Y9 25131876 Ki = 27.54 nM T92609 CNQX42 25132217 Ki > 1000 nM T92609 C7WE4Y 25132564 Ki = 512.86 nM T92609 C6K1TB 25132565 Ki = 407.38 nM T92609 CJ19KC 25132566 Ki = 87.1 nM T92609 C79CVE 25154770 EC50 = 658 nM T92609 CNO83H 25181488 Ki = 16.6 nM T92609 CEYF08 25181489 Ki = 128.82 nM T92609 CAM63X 42618195 IC50 > 1000 nM T92609 C8K4UF 42618197 IC50 > 1000 nM T92609 CY7W2J 42631003 Ki = 19.05 nM T92609 CJ3NP5 42636941 IC50 = 74.13 nM T92609 CW2DP3 44123711 Ki = 91.2 nM T92609 CJ41QV 44126269 Ki = 7.079 nM T92609 C2HPM1 44213730 Ki = 7.943 nM T92609 C2DS9L 44213782 Ki = 3 nM T92609 CTR42S 44219718 EC50 = 1 nM T92609 CB2HY8 44219719 EC50 = 51 nM T92609 C76ONX 44219756 IC50 > 10000 nM T92609 C4T7ZI 44222842 Ki = 81.28 nM T92609 C9ROX7 44267817 Ki = 83 nM T92609 C0L4TU 44267884 Ki = 38 nM T92609 CF2DH7 44267890 Ki = 129 nM T92609 CEL7U6 44267912 Ki = 98 nM T92609 CF51JW 44268966 Ki = 8.49 nM T92609 C89FEL 44269124 EC50 = 3.162 nM T92609 CVE83T 44271661 EC50 = 0.7943 nM T92609 C7P2AH 44271931 EC50 = 251.19 nM T92609 CSQ5L6 44271932 EC50 = 6.31 nM T92609 C5UA4W 44273916 Ki = 4.8 nM T92609 CMH52E 44275255 Ki = 1.259 nM T92609 C1SZ4H 44275505 Ki = 0.36 nM T92609 C7Q2JD 44275526 Ki = 69.18 nM T92609 CK2R3A 44276536 Ki = 963 nM T92609 CA0DZ5 44280965 EC50 = 30000 nM T92609 C2TNR1 44280982 EC50 = 340 nM T92609 C9KVJ2 44281057 EC50 = 5300 nM T92609 CA15SP 44281250 EC50 = 200 nM T92609 C03CBT 44281493 EC50 = 170 nM T92609 CN5YC0 44281507 EC50 = 30000 nM T92609 CPK7B3 44284333 Ki = 33.88 nM T92609 CZPD80 44288485 Ki = 5.1 nM T92609 C5UIM4 44288492 Ki = 380 nM T92609 CL3RI0 44288729 Ki = 42 nM T92609 CTR4Z6 44288740 Ki = 28 nM T92609 C4K6RC 44288741 Ki = 74 nM T92609 CQP9B7 44288754 Ki = 47 nM T92609 CZ5P6U 44288769 Ki = 1.1 nM T92609 CV8G1J 44288792 Ki = 6.4 nM T92609 CQ40MA 44288794 Ki = 50 nM T92609 CX7BT8 44288810 Ki = 570 nM T92609 CA16JS 44288815 Ki = 7.4 nM T92609 C4KND2 44288816 Ki = 61 nM T92609 CT7IB6 44288841 Ki = 8.8 nM T92609 CEM2T4 44288843 Ki = 13 nM T92609 CZ7O4D 44288847 Ki = 1.4 nM T92609 C8EJ9B 44288857 Ki = 75 nM T92609 CKA01M 44288858 Ki = 3.2 nM T92609 CL4X9R 44288864 Ki = 257 nM T92609 C6DYQ1 44288874 Ki = 1 nM T92609 CAG7E1 44288877 Ki = 7 nM T92609 CQ74LV 44288917 Ki = 1.8 nM T92609 CQ3Y5R 44288945 Ki = 0.4 nM T92609 CZDR39 44288995 Ki = 24 nM T92609 C92FEY 44289026 Ki = 22 nM T92609 C9HMK3 44289034 Ki = 3.4 nM T92609 C5ZL4A 44289035 Ki = 1.9 nM T92609 C71XMR 44289047 Ki = 27 nM T92609 CW5C4G 44289058 Ki = 72 nM T92609 C62NWB 44289089 Ki = 240 nM T92609 C37GEA 44289100 Ki = 0.7 nM T92609 C1ES5Y 44289103 Ki = 3 nM T92609 CZS9B7 44289107 Ki = 1 nM T92609 CZSM05 44289112 Ki = 7.5 nM T92609 C51NLQ 44289248 Ki = 0.08913 nM T92609 CWC49F 44289261 Ki = 0.5129 nM T92609 C14WMG 44289321 Ki = 1.1 nM T92609 CQW1Z3 44289344 Ki = 12 nM T92609 CFO29U 44289346 Ki = 25 nM T92609 C1JX5M 44289437 Ki = 0.2512 nM T92609 CIM92E 44289525 Ki = 4.1 nM T92609 CF1UW9 44294569 Ki = 4.75 nM T92609 CBS42M 44294957 Ki = 0.6 nM T92609 CW6D7V 44294958 Ki = 2.3 nM T92609 CR9K8P 44295016 Ki < 1 nM T92609 CMQ6G5 44295044 Ki = 5.8 nM T92609 C9XAB7 44295046 Ki = 1.1 nM T92609 C9MQ4B 44295133 Ki = 9.1 nM T92609 CNQ82T 44295170 Ki = 62 nM T92609 C9Y3GE 44295192 Ki = 0.9 nM T92609 C4KB8E 44295193 Ki = 35 nM T92609 C9UW2H 44295218 Ki = 15 nM T92609 CWJ13T 44298447 Ki = 0.5012 nM T92609 C0F8LH 44298611 Ki = 0.03981 nM T92609 C0M5BZ 44298624 Ki = 0.1585 nM T92609 C17AXP 44298626 Ki = 0.3162 nM T92609 CA19EZ 44298644 Ki = 3.981 nM T92609 C0QLW1 44298650 Ki = 0.2512 nM T92609 CO6K1V 44298664 Ki = 0.0631 nM T92609 CMI12L 44298671 Ki = 1.585 nM T92609 CBJ31S 44298694 Ki = 1.995 nM T92609 CUO47C 44298734 Ki = 1.585 nM T92609 CDLJ86 44298735 Ki = 2.512 nM T92609 C4N1EM 44298746 Ki = 0.7943 nM T92609 C1V0RE 44298747 Ki = 19.95 nM T92609 C1H2MT 44298762 Ki = 6.31 nM T92609 C3X6RY 44298770 Ki = 1 nM T92609 C9TR2K 44298780 Ki = 5.012 nM T92609 CX90HD 44299835 Ki = 4.7 nM T92609 C6HO4W 44299945 Ki = 2.3 nM T92609 CG82KA 44299973 Ki = 0.9 nM T92609 CL62DY 44299974 Ki = 0.44 nM T92609 C0LF1S 44299975 Ki = 1.6 nM T92609 CY8J6F 44300087 Ki = 0.46 nM T92609 CYV46S 44300107 Ki = 0.6 nM T92609 CLHT17 44300111 Ki = 0.4 nM T92609 C2WP7S 44300129 Ki = 0.38 nM T92609 CH59JV 44300159 Ki = 2.4 nM T92609 C8K3AP 44300165 Ki = 0.24 nM T92609 CSA23P 44300166 Ki = 8.3 nM T92609 C3YDV9 44300170 Ki = 2.4 nM T92609 CW56GZ 44301572 Ki = 220 nM T92609 CH34AY 44301573 Ki = 9.7 nM T92609 CIPQ70 44301680 Ki = 77 nM T92609 C5EZ6B 44301681 Ki = 5.7 nM T92609 C6R2DV 44308443 Ki = 18 nM T92609 C8M4HW 44308466 Ki = 12 nM T92609 CPUO39 44308654 Ki = 419 nM T92609 CB18TU 44309199 Ki = 7300 nM T92609 C6G8ZC 44311789 Ki = 14125.38 nM T92609 C5L1WN 44312036 Ki < 100000 nM T92609 CT46CK 44312037 Ki = 21379.62 nM T92609 C3XFH4 44312198 Ki = 91201.08 nM T92609 CZ4TN0 44314198 Ki = 141.25 nM T92609 CCI07K 44314200 Ki = 1949.84 nM T92609 CKU7Y6 44316072 Ki = 9 nM T92609 CG2UB8 44316098 Ki = 3.7 nM T92609 C2PR8V 44318000 Ki = 82 nM T92609 CZ5M4K 44318075 Ki = 86 nM T92609 C8JKO2 44318081 Ki = 100 nM T92609 CV8WZ0 44318454 IC50 = 44.67 nM T92609 CXJL56 44318842 IC50 = 42.66 nM T92609 C3J9XH 44324405 Ki = 0.068 nM T92609 CGP40I 44329083 EC50 < 5011.87 nM T92609 CES26R 44329133 EC50 = 79.43 nM T92609 CR3N5S 44329318 EC50 < 5011.87 nM T92609 CZ21VE 44329481 EC50 = 19.95 nM T92609 C4ZV9T 44329701 EC50 = 501.19 nM T92609 CBZ84S 44329703 EC50 = 7.943 nM T92609 CQY03V 44329738 EC50 < 5011.87 nM T92609 C7Z2HM 44329739 EC50 = 39.81 nM T92609 CS2WN0 44329788 EC50 = 1.259 nM T92609 C5AG1U 44329790 EC50 = 12.59 nM T92609 C14RBX 44329796 EC50 = 10 nM T92609 CG60QK 44329797 EC50 = 3.162 nM T92609 C6US9E 44330880 Ki = 45 nM T92609 C2N0GV 44331079 Ki = 71 nM T92609 C02JUQ 44331090 Ki = 20 nM T92609 CU2H1F 44331136 Ki = 13 nM T92609 C5SLE2 44331150 Ki = 8 nM T92609 CK5R0A 44331169 Ki = 6.5 nM T92609 CGJB37 44331174 Ki = 31 nM T92609 CI9UV3 44331198 Ki = 56 nM T92609 C4RJ7I 44331277 Ki = 53 nM T92609 CO5T9G 44343173 EC50 = 63.1 nM T92609 C0DS6V 44343235 EC50 = 158.49 nM T92609 CK1QJ5 44343236 EC50 = 6.31 nM T92609 CV5N1T 44343243 EC50 = 63.1 nM T92609 C84GDJ 44343244 EC50 = 6.31 nM T92609 CV8LE9 44343245 EC50 = 50.12 nM T92609 CX8J0Y 44343247 EC50 = 3.981 nM T92609 C71WZX 44343251 EC50 = 125.89 nM T92609 C19JFN 44343257 EC50 = 15.85 nM T92609 C17HRU 44343275 EC50 = 50.12 nM T92609 C6ZU5G 44343410 EC50 = 10 nM T92609 CQR12J 44343520 EC50 < 5011.87 nM T92609 CFQ32B 44343524 EC50 < 100000 nM T92609 C6N3XK 44345317 IC50 < 1000 nM T92609 CZ2X3A 44352155 EC50 = 7.943 nM T92609 C3I9DE 44358574 Ki = 0.55 nM T92609 C2WYI7 44361064 Ki = 95.5 nM T92609 C8OM7A 44362013 EC50 = 158.49 nM T92609 CK6S1Y 44362145 EC50 = 100 nM T92609 C7FHB4 44362146 EC50 = 0.2512 nM T92609 CSFJ14 44362149 EC50 = 5.012 nM T92609 CEZ8K0 44362150 EC50 = 5.012 nM T92609 CK8U9S 44362185 EC50 = 1.995 nM T92609 CHL40X 44362194 EC50 = 0.5012 nM T92609 C3CF8S 44362195 EC50 = 1.259 nM T92609 C78CEY 44362196 EC50 = 2.512 nM T92609 C3AU6V 44362208 EC50 = 1 nM T92609 CH9B3A 44362286 EC50 = 1.259 nM T92609 CF6H7S 44362287 EC50 < 100000 nM T92609 CI6DH4 44362288 EC50 = 2.512 nM T92609 C2SBP1 44362289 EC50 = 1258.93 nM T92609 CH79ZL 44362510 EC50 = 125.89 nM T92609 C0GR4S 44362511 IC50 = 1288.25 nM T92609 C1U0TR 44362523 EC50 < 100000 nM T92609 CEQD62 44362541 EC50 < 100000 nM T92609 CU0E7G 44362633 Ki = 4.2 nM T92609 C94ORM 44362867 Ki = 4.6 nM T92609 CZ1KQ9 44369351 EC50 = 2.239 nM T92609 C1Y7OL 44369431 EC50 = 0.8511 nM T92609 C03STZ 44369434 EC50 = 2.692 nM T92609 C6W2MT 44369646 EC50 = 36.31 nM T92609 CDR8C3 44369647 EC50 = 45.71 nM T92609 C3K6GE 44376845 IC50 = 5248.07 nM T92609 CPD18R 44376900 IC50 = 245.47 nM T92609 CE46SW 44376923 IC50 = 398.11 nM T92609 C7UW8Z 44376927 IC50 = 5888.44 nM T92609 C8GT5O 44376936 IC50 = 812.83 nM T92609 CLC2T4 44376954 IC50 = 239.88 nM T92609 C9IPC3 44376958 IC50 = 112.2 nM T92609 CX4A1Z 44376975 IC50 = 204.17 nM T92609 C14SMK 44376984 IC50 = 478.63 nM T92609 C0V4XL 44376993 IC50 = 2570.4 nM T92609 CB2R0M 44377007 IC50 = 281.84 nM T92609 C2ID6U 44377035 IC50 = 691.83 nM T92609 C6R9OZ 44377036 IC50 = 724.44 nM T92609 C97QIG 44377200 IC50 = 891.25 nM T92609 CUG3H0 44388493 Ki = 300 nM T92609 C1H9EK 44388495 Ki = 9.5 nM T92609 CBP8H3 44390704 Ki = 20 nM T92609 COFG53 44390739 Ki = 0.2 nM T92609 C6YP8T 44404321 Ki = 5.25 nM T92609 CYA37J 44404326 Ki = 5.25 nM T92609 C27FZA 44417706 Ki = 33.88 nM T92609 C31WOV 44417713 Ki = 4.571 nM T92609 C85GUJ 44420408 Ki = 8.318 nM T92609 CHIA46 44420412 Ki = 53.7 nM T92609 C6I3MN 44420418 Ki = 4265.8 nM T92609 CQV5N7 44420419 Ki = 181.97 nM T92609 CSQ5H2 44420423 Ki = 30.2 nM T92609 C1CFB6 44420428 Ki = 1.479 nM T92609 CAW15U 44420431 Ki = 3.467 nM T92609 C7C4QE 44426404 Ki = 14 nM T92609 CE3XQ2 44426405 Ki = 5.4 nM T92609 C21KYB 44428845 Ki = 3.467 nM T92609 C91BHJ 44428846 Ki = 27.54 nM T92609 CCLI02 44428847 Ki = 25.7 nM T92609 CE08JS 44428848 Ki = 4.266 nM T92609 CVH1Z5 44428849 Ki = 10.47 nM T92609 CY26IH 44428850 Ki = 48.98 nM T92609 CRN18J 44428851 Ki = 4.169 nM T92609 CBK87I 44431173 Ki = 37.8 nM T92609 CX3D0B 44431174 Ki = 2.7 nM T92609 C9HD0G 44431180 Ki = 1.8 nM T92609 CB3A8T 44431184 Ki = 3.9 nM T92609 C09VIB 44431192 Ki = 0.8 nM T92609 C43SCL 44431194 Ki = 0.4 nM T92609 C4G7QF 44431545 Ki = 2.7 nM T92609 C8OP5V 44431546 Ki = 0.77 nM T92609 C0B5TC 44431547 Ki = 0.88 nM T92609 CCXB24 44431548 Ki = 1 nM T92609 C5QI0V 44431551 Ki = 0.73 nM T92609 C2R4TP 44431553 Ki = 14 nM T92609 COIS42 44431554 Ki = 1.3 nM T92609 C0APQ4 44431555 Ki = 4.8 nM T92609 CJT34W 44431557 Ki = 17 nM T92609 CF76RP 44431560 Ki = 1.6 nM T92609 CY8C0V 44431562 Ki = 8.7 nM T92609 C2UD6M 44431564 Ki = 0.9 nM T92609 C4J0TG 44431574 Ki = 6 nM T92609 C0C8TU 44431587 Ki = 1.6 nM T92609 C1QV6S 44431590 Ki = 25 nM T92609 CF3ST7 44431594 Ki = 1 nM T92609 CA9O2E 44431599 Ki = 1.5 nM T92609 CX9YA2 44431602 Ki = 1.6 nM T92609 C9OSE8 44431607 Ki = 0.56 nM T92609 CT0LP1 44431611 Ki = 3 nM T92609 C46NHX 44431612 Ki = 45 nM T92609 C3IA4W 44431613 Ki = 189 nM T92609 C5QJ8S 44431614 Ki = 19 nM T92609 CXD1Q9 44431615 Ki = 36 nM T92609 C0WPS6 44431616 Ki = 1.2 nM T92609 C4SZA3 44431617 Ki = 5 nM T92609 CE6L0D 44431618 Ki = 4.9 nM T92609 CS9N3Q 44431620 Ki = 3.5 nM T92609 CEWQ41 44433348 Ki = 15 nM T92609 CZ3RM2 44435219 Ki = 330 nM T92609 C64POV 44449245 EC50 = 52 nM T92609 CX7Z6I 44449247 EC50 = 167 nM T92609 CO9NC7 44449248 EC50 = 451 nM T92609 C1P3XZ 44449249 EC50 = 33 nM T92609 CN9BI4 44449276 EC50 = 2200 nM T92609 CYM30S 44449277 EC50 = 32 nM T92609 CS5WB3 44449278 EC50 = 142 nM T92609 CH74NV 44449303 EC50 = 78 nM T92609 C8VO6A 44449304 EC50 = 70 nM T92609 CI4T2K 44449305 EC50 = 32 nM T92609 C70SEG 44449306 EC50 = 1340 nM T92609 C0M7UN 44449337 EC50 = 322 nM T92609 C4THN7 44449338 EC50 = 473 nM T92609 C1O6QI 44449657 EC50 = 111 nM T92609 C6QCN8 44449686 EC50 = 426 nM T92609 CH5RL7 44449690 EC50 = 1150 nM T92609 CS3LB0 44449691 EC50 = 2060 nM T92609 CFL25O 44449692 EC50 = 170 nM T92609 CSZB25 44449694 EC50 > 1300 nM T92609 CJ8WL7 44449723 EC50 = 278 nM T92609 C8XHB5 44449724 EC50 > 2900 nM T92609 C6ZG3O 44449725 EC50 = 3 nM T92609 CMLE59 44449730 EC50 = 14 nM T92609 C12XGE 44456400 Ki > 10000 nM T92609 CGO23X 44460394 Ki = 1298 nM T92609 CLVD72 44460423 Ki = 15 nM T92609 C7T2KE 44460449 Ki = 3466 nM T92609 CVJ72X 44460477 Ki = 28 nM T92609 CT5M7N 44460522 Ki = 297 nM T92609 CV3IW1 44461012 Ki = 90 nM T92609 CQ2IX7 44461606 IC50 = 1905.46 nM T92609 C1PI3F 44462130 Ki = 44 nM T92609 CJ10OZ 44531812 Ki = 194.98 nM T92609 CT85QK 44538690 Ki = 262 nM T92609 CT9S4L 44563063 IC50 = 2400 nM T92609 CDTB89 44563137 IC50 > 10000 nM T92609 CAR23X 44568818 Ki = 223.87 nM T92609 CAO31F 44568917 Ki = 74.13 nM T92609 CE3GV8 44568918 Ki = 89.13 nM T92609 CN34AO 44571840 EC50 = 84 nM T92609 CVO6K5 44571841 EC50 = 37 nM T92609 CBV05O 44571842 EC50 = 62 nM T92609 CEZC45 44571843 EC50 = 168 nM T92609 CR07VH 44571844 EC50 = 195 nM T92609 CZ5H1K 44571845 EC50 = 879 nM T92609 C13ZGP 44571887 EC50 = 62 nM T92609 C5C3RV 44571888 EC50 = 59 nM T92609 CO63WS 44571889 EC50 = 32 nM T92609 C2TWZ8 44571890 EC50 = 90 nM T92609 C7Z8SC 44571891 EC50 = 111 nM T92609 CMUP18 44571937 EC50 = 17 nM T92609 C5CRY0 44571938 Ki = 5 nM T92609 C81IMZ 44573820 IC50 = 350 nM T92609 CEF6J8 44573821 IC50 = 230 nM T92609 CT2FW6 44573822 IC50 = 470 nM T92609 C4I5UB 44573823 IC50 = 920 nM T92609 CXWQ34 44573931 IC50 = 3600 nM T92609 C6U0EY 44573932 IC50 = 1910 nM T92609 C04SIR 44573964 IC50 = 1160 nM T92609 CAT49R 44574008 IC50 > 10000 nM T92609 CVF30Y 44574044 EC50 = 51 nM T92609 CCD72N 44574045 EC50 = 12 nM T92609 CMS20J 44574074 EC50 = 0.4 nM T92609 C92YUA 44574075 EC50 = 2 nM T92609 C9NU2C 44574076 EC50 = 92 nM T92609 CB8US6 44574077 EC50 = 3 nM T92609 CX4Y0K 44574078 EC50 = 1 nM T92609 CU9X8G 44574079 EC50 = 81 nM T92609 C62FCK 44574080 EC50 = 9 nM T92609 CAT57X 44574103 EC50 = 5 nM T92609 CXZ0J3 44574104 EC50 = 4 nM T92609 CES4X0 44574105 EC50 = 12 nM T92609 C62AYR 44574106 EC50 = 19 nM T92609 CX98MY 44574107 EC50 = 19 nM T92609 CDER54 44574132 EC50 = 62 nM T92609 C4S2OQ 44574133 EC50 = 33 nM T92609 C96NQZ 44574134 EC50 = 3 nM T92609 CKR69S 44574135 EC50 = 15 nM T92609 C4WZG9 44574136 EC50 = 3 nM T92609 CL37FD 44574137 EC50 = 5 nM T92609 CG0RM2 44574138 EC50 = 27 nM T92609 C0VQ8Y 44574357 IC50 = 340 nM T92609 CQZ1Y2 44574358 IC50 = 540 nM T92609 C0SOD6 44574359 IC50 = 490 nM T92609 CD87ZE 44574834 EC50 = 1650 nM T92609 C2YF8O 44574874 EC50 = 276 nM T92609 CFQJ71 44574875 EC50 = 514 nM T92609 CB1R3O 44574876 EC50 > 10000 nM T92609 CR8SF7 44574877 EC50 = 144 nM T92609 CN94EW 44574878 EC50 = 1050 nM T92609 C8L6CN 44574934 EC50 > 10000 nM T92609 CVN8Z4 44574935 EC50 = 19 nM T92609 C9QAM5 44574936 EC50 = 3460 nM T92609 CHT2Z9 44574937 EC50 = 22 nM T92609 CV06SB 44574938 EC50 = 578 nM T92609 CU4M3D 44574985 EC50 = 939 nM T92609 C3QWO0 44574986 EC50 = 42 nM T92609 C3GC6T 44574987 EC50 = 11 nM T92609 C4GQR8 44574988 EC50 = 371 nM T92609 C4XHI5 44574989 EC50 = 82 nM T92609 CYAI96 44575544 IC50 = 13 nM T92609 CRCH48 44582675 Ki = 335 nM T92609 CEJ4R8 44582676 Ki = 146 nM T92609 C9F6EB 44593557 EC50 = 27 nM T92609 C51AJZ 44593577 EC50 = 123 nM T92609 CDA54Q 44593580 EC50 = 48 nM T92609 C1SN7Y 44593709 Ki = 18.62 nM T92609 CWO70X 45260703 EC50 = 489.78 nM T92609 C4VOW6 45260704 EC50 = 5.012 nM T92609 CQ0R5Y 45264581 EC50 = 4.571 nM T92609 C39CDN 45264638 EC50 = 3.388 nM T92609 C0F4TJ 45268939 Ki = 2.818 nM T92609 CM5H4D 45280021 EC50 > 10000 nM T92609 CPJB52 45280075 EC50 = 1548 nM T92609 CMNA70 45358442 Ki = 158.49 nM T92609 CV0JK1 45380469 EC50 = 1757 nM T92609 C6QES8 45380471 EC50 > 10000 nM T92609 CZ73IE 45381852 EC50 = 857 nM T92609 CNI72R 45381932 EC50 > 10000 nM T92609 C8WG5T 45381933 EC50 = 812 nM T92609 CGLF37 45484995 IC50 = 3600 nM T92609 CGOS24 45485061 IC50 = 1320 nM T92609 CLX9C8 45485062 IC50 = 2790 nM T92609 C05PBD 46176231 IC50 > 10000 nM T92609 C2L5UH 46182745 IC50 = 8150 nM T92609 C5FQ4S 46224879 Ki = 1.413 nM T92609 C0ABR3 46846073 Ki = 489.78 nM T92609 C03LTM 46869265 Ki = 340000 nM T92609 C7ZEI6 46881382 Ki = 35.48 nM T92609 CN0Q2A 46881443 Ki = 91.2 nM T92609 CGX02N 46881444 Ki = 48.98 nM T92609 C4U6RH 46881493 Ki = 117.49 nM T92609 CV7R9S 46881494 Ki = 20.89 nM T92609 C24QFO 46882032 Ki > 1000 nM T92609 C3GQW6 46882033 Ki > 1000 nM T92609 CPG6U5 46882034 Ki = 2.089 nM T92609 CYB37P 46882085 Ki = 6.607 nM T92609 CD8CX3 46882086 Ki = 302 nM T92609 C57GAO 46882087 Ki > 1000 nM T92609 CV3QW9 46882088 Ki = 85.11 nM T92609 C5ZDY3 46915370 Ki = 885 nM T92609 CI4XZ1 46934637 Ki = 11.48 nM T92609 CK1Z0M 46934639 Ki = 0.871 nM T92609 CU0TB9 46934641 Ki = 26.92 nM T92609 CR6JV7 46934643 Ki = 0.631 nM T92609 C14ZLO 46934645 Ki = 40.74 nM T92609 C2N9JZ 46934787 Ki = 2.884 nM T92609 CI4U0L 46934789 Ki = 21.38 nM T92609 C8HVG6 46934791 Ki = 6.607 nM T92609 CA51JI 46934793 Ki = 10 nM T92609 CB4Z7D 46934945 Ki = 2.042 nM T92609 C2LZJ0 49783209 Ki = 522 nM T92609 C57SMG 49783415 Ki > 10000 nM T92609 C0TG6I 49783419 Ki = 87.6 nM T92609 C0D5GI 49796077 Ki = 831.76 nM T92609 C6ZRD7 49797187 Ki = 102.33 nM T92609 C63FGJ 49797190 Ki = 100 nM T92609 C6IW4Q 49862238 Ki = 76 nM T92609 CZ2SA8 49864841 Ki = 3.981 nM T92609 C8J5PI 49865599 Ki = 23 nM T92609 CP63AX 49865600 Ki = 33 nM T92609 CA1IY0 49865601 Ki = 593 nM T92609 CC5KD7 49865639 Ki = 17 nM T92609 C1B5RD 49865640 Ki = 14 nM T92609 C51PJT 49865641 Ki = 40 nM T92609 C3KF6B 49865668 Ki = 6 nM T92609 C2RY0J 50878551 Ki > 10000 nM T92609 C1W6TV 50898777 Ki > 10000 nM T92609 CXMZ73 50898778 Ki > 10000 nM T92609 C8EU7J 50905381 Ki = 0.3388 nM T92609 CW7FI3 50905585 Ki = 0.3467 nM T92609 CIL56G 50905588 Ki = 19.05 nM T92609 C5M6VO 50905589 Ki = 11.48 nM T92609 CE4KP1 51050257 Ki > 10000 nM T92609 CJ9L0W 51347282 EC50 = 1250 nM T92609 CQG7X2 51349173 EC50 > 10000 nM T92609 CF9V1U 52937018 Ki = 316.23 nM T92609 CS3BJ7 52937119 Ki = 100 nM T92609 C93QXP 52937222 Ki = 15.85 nM T92609 CPF7V0 52937223 Ki = 316.23 nM T92609 CYG24L 52937526 Ki = 125.89 nM T92609 CL8QZ3 52937527 Ki = 251.19 nM T92609 CM36PE 52937629 Ki = 794.33 nM T92609 CRV61I 52937630 Ki = 63.1 nM T92609 CEKB47 52937631 Ki = 10 nM T92609 CZ0C5B 52937632 Ki > 1995.26 nM T92609 CVX7U2 52937633 Ki > 1995.26 nM T92609 C3ZX1Q 52937634 Ki > 1995.26 nM T92609 CY4N8T 52937728 Ki = 50.12 nM T92609 C83WTP 52937729 Ki = 398.11 nM T92609 CQDS92 52937730 Ki = 1584.89 nM T92609 CR0KW9 52937731 Ki = 501.19 nM T92609 C2UV5S 52937732 Ki = 199.53 nM T92609 C6XHP8 52937733 Ki > 1995.26 nM T92609 C3B5HN 52937734 Ki > 1995.26 nM T92609 CK52QG 52937828 Ki = 199.53 nM T92609 CFV4D0 52937829 Ki = 501.19 nM T92609 C9MBQ2 52937830 Ki = 39.81 nM T92609 CLW3B0 52940951 Ki = 2.512 nM T92609 CWYS78 52941004 Ki = 1.995 nM T92609 CE0X9W 52941056 Ki = 10 nM T92609 C40WVE 52941624 Ki = 3.162 nM T92609 CV7HZ6 52942047 Ki = 1.38 nM T92609 C5Y3VS 52942152 Ki = 1.122 nM T92609 CO9J6M 52943356 Ki = 2.512 nM T92609 CRL3P0 52944615 Ki = 6.31 nM T92609 C4N6ET 52944674 Ki = 5.012 nM T92609 CDQ27E 52945156 Ki = 19.95 nM T92609 CPI9F4 52945803 Ki = 3.162 nM T92609 CGZ1R7 52947088 Ki = 7.943 nM T92609 CNH57S 52947579 Ki = 3.162 nM T92609 CX04NC 52948119 Ki = 12.59 nM T92609 C9YBJ3 52948823 Ki = 9.772 nM T92609 CCQZ15 52949448 Ki = 0.263 nM T92609 CGY45S 53248361 Ki = 78 nM T92609 CE9L8G 53248365 Ki = 176 nM T92609 C4H5JI 53327748 Ki = 1.82 nM T92609 C1YX4A 53327991 Ki = 22.39 nM T92609 CUP50Y 53327992 Ki = 9.772 nM T92609 CZ1B6D 53328115 Ki = 3467.37 nM T92609 CT0D9O 53328116 Ki = 3235.94 nM T92609 CGB3U6 53328311 Ki = 46.77 nM T92609 CIWJ61 53328312 Ki = 47.86 nM T92609 CW36HN 53328313 Ki = 190.55 nM T92609 C6NUW4 53328314 Ki = 15.85 nM T92609 C7XCQ4 53328315 Ki = 36.31 nM T92609 CJ7TY9 53328316 Ki = 21.88 nM T92609 C76NJW 53328503 Ki = 1698.24 nM T92609 CB1D8L 53328504 Ki = 6918.31 nM T92609 CY9JI7 53328505 Ki = 28.18 nM T92609 C5FHA1 53328506 Ki = 48.98 nM T92609 CCM7S9 53328507 Ki = 67.61 nM T92609 C7YN2M 53328508 Ki = 14.13 nM T92609 CD7EB0 53328684 Ki = 20.89 nM T92609 CQGE30 53328685 Ki = 10.23 nM T92609 CNSU94 53328686 Ki = 34.67 nM T92609 CY51RC 53328687 Ki = 95.5 nM T92609 C9L0ZI 53328872 Ki = 3388.44 nM T92609 C67YNQ 53328873 Ki = 63.1 nM T92609 CGX1W2 53779053 Ki = 13 nM T92609 C6W1RA 56649648 Ki = 16 nM T92609 C2SW7J 56649649 Ki = 74 nM T92609 CQTR49 56649650 Ki = 36 nM T92609 CA6B2I 56668277 Ki = 1 nM T92609 CU0NE5 56672197 Ki > 10000 nM T92609 CJKO58 56852956 Ki = 257.04 nM T92609 CB0P9N 56944383 Ki = 0.8 nM T92609 CCW38Z 56945164 Ki = 109.65 nM T92609 CN6XE8 56945165 Ki = 38.9 nM T92609 CPE6C7 56945166 Ki > 1000 nM T92609 C4L7GW 56945167 Ki = 44.67 nM T92609 CL68PZ 56946472 Ki = 53.7 nM T92609 CJ98DO 56946474 Ki = 26.92 nM T92609 CB8J2F 56946573 Ki = 0.6457 nM T92609 CCBY53 56946575 Ki > 1000 nM T92609 CMO0U3 56946577 Ki > 1000 nM T92609 CJZ3P4 56946579 Ki = 39.81 nM T92609 CXUW26 56961460 Ki = 2.1 nM T92609 CX74AS 56961506 Ki = 1.3 nM T92609 C9WP3O 56961507 Ki = 4.7 nM T92609 C1TC7Q 56963799 Ki > 10000 nM T92609 CDTG05 57393527 Ki = 0.263 nM T92609 CR1Y7M 57398332 Ki > 10000 nM T92609 C8EFT7 57402251 Ki > 1000 nM T92609 CT89JH 57780007 Ki = 251.19 nM T92609 CT8RO7 57780008 Ki = 7.943 nM T92609 C5RIN4 57780016 Ki = 63.1 nM T92609 CE9WC0 57780017 Ki > 1995.26 nM T92609 C1W4SB 57780018 Ki > 1995.26 nM T92609 CT96WD 57780020 Ki = 316.23 nM T92609 C2PJ4N 59271992 IC50 = 500 nM T92609 C7WL6M 68155065 EC50 > 10000 nM T92609 C1SBP9 69781970 Ki = 5.495 nM T92609 CCD2L1 69782867 Ki = 0.871 nM T92609 CC43QK 71151588 Ki = 16.9 nM T92609 CBQ8P4 71449250 Ki = 19.95 nM T92609 C6SN2P 71449516 Ki = 66.07 nM T92609 C6DU5P 71450548 Ki > 10000 nM T92609 C9VZ8J 71450550 Ki = 472 nM T92609 CFS69A 71450901 Ki = 31.62 nM T92609 CB83YL 71451044 Ki = 100 nM T92609 C6ZWV2 71452383 Ki > 10000 nM T92609 CDTW09 71452387 Ki > 10000 nM T92609 C75EQJ 71452768 Ki = 0.9 nM T92609 C0YXD3 71452871 Ki = 12.59 nM T92609 CY7NM9 71452872 Ki = 630.96 nM T92609 C4JN5I 71454639 Ki = 50.12 nM T92609 C31VFN 71454865 Ki = 2.188 nM T92609 C8YH0J 71455083 Ki = 39 nM T92609 C6G2HC 71455894 Ki > 10000 nM T92609 CMBU21 71456359 Ki = 19.95 nM T92609 CVT39B 71456360 Ki = 316.23 nM T92609 CK87DI 71456361 Ki = 398.11 nM T92609 CP7JI0 71457691 Ki > 10000 nM T92609 C3VMS0 71458203 Ki = 12.59 nM T92609 C8T5EJ 71458204 Ki = 199.53 nM T92609 CZ6BX7 71458205 Ki = 158.49 nM T92609 CORB94 71458492 Ki = 5.623 nM T92609 CEBC62 71461781 Ki = 15.85 nM T92609 C9DJ1V 71461782 Ki = 6.31 nM T92609 CA6NI7 71462043 Ki = 0.8913 nM T92609 CD9G8B 71521478 Ki > 1000 nM T92609 CSV0G5 71521479 Ki = 257.04 nM T92609 CGN2M7 71521480 Ki = 436.52 nM T92609 CDS15J 71659980 Ki = 1.122 nM T92609 CI0GU8 71660496 IC50 > 48500 nM T92609 C8QO1W 71719108 Ki = 360 nM T92609 CH6J4G 71817545 Ki = 177.83 nM T92609 CH54DW 71817546 Ki = 1.995 nM T92609 C3NO8R 71817548 Ki = 3.802 nM T92609 CRTD80 71817857 Ki = 436.52 nM T92609 CBTX18 71817858 Ki = 16.98 nM T92609 CRYP87 71817860 Ki = 31.62 nM T92609 C3ATN5 72197484 IC50 = 1390 nM T92609 CN8A5R 72197486 IC50 > 10000 nM T92609 CC65OA 73213195 Ki > 10000 nM T92609 CW83DK 73213196 Ki = 286 nM T92609 CCV91B 73346042 Ki = 21.4 nM T92609 CK0HR9 73346334 Ki = 6085 nM T92609 CY60RD 73347826 Ki = 2276 nM T92609 CX01MD 73349178 Ki = 9.12 nM T92609 C8GQK9 73350823 Ki = 80 nM T92609 CAI63V 73355417 Ki > 10000 nM T92609 CBW1D8 73356785 Ki = 0.4898 nM T92609 CVF5P0 73603034 IC50 = 2500 nM T92609 C2E7QW 75201901 Ki = 3400 nM T92609 C8IDL3 75306277 Ki = 501.19 nM T92609 CFN6P8 76071738 IC50 = 57.4 nM T92609 CW61JI 76071739 IC50 = 12.8 nM T92609 C1L3CT 76071859 IC50 = 3187 nM T92609 CX57RZ 76307950 Ki = 36.3 nM T92609 C1G4EZ 76307951 Ki = 1698.2 nM T92609 CV24YC 76307952 Ki = 223.87 nM T92609 C04HNK 76308473 Ki = 27.54 nM T92609 CE34XR 76311538 Ki = 407.38 nM T92609 C7EFN8 76311539 Ki = 537.03 nM T92609 C7Q8MV 76315111 Ki = 0.08 nM T92609 C5V6EL 76318762 Ki = 338.84 nM T92609 CQ24UF 76318763 Ki = 95.49 nM T92609 CMG38P 76318764 Ki = 467.74 nM T92609 CDY1W7 76322411 Ki = 169.82 nM T92609 CEB54F 76322412 Ki = 28.84 nM T92609 CD0UV1 76322413 Ki = 512.86 nM T92609 C8M3OX 76323009 Ki = 23.44 nM T92609 CS02IK 76326030 Ki = 7.94 nM T92609 COT51G 76326561 Ki = 25.7 nM T92609 CFV87U 76330228 Ki = 3.467 nM T92609 CP3D9T 76333279 Ki = 0.05 nM T92609 C6A2RT 76333280 Ki = 2.34 nM T92609 C92VJX 76333281 Ki = 158.49 nM T92609 C7WRV3 76333282 Ki = 74.13 nM T92609 C3Z1TP 78815633 Ki = 1.122 nM T92609 CL9AI7 85469698 IC50 = 151.3 nM T92609 CGO74F 85469753 IC50 = 3421 nM T92609 C91LTS 85469754 IC50 = 46.44 nM T92609 CS9DG8 85469755 IC50 = 89.94 nM T92609 CU6R1L 85469756 IC50 = 884.7 nM T92609 CTRN10 85469757 IC50 = 128 nM T92609 CU3P0H 85469808 IC50 = 1200 nM T92609 C74PRV 85469809 IC50 = 14.25 nM T92609 CUOH37 85469811 IC50 = 15.16 nM T92609 CKNG20 85469812 IC50 = 32.43 nM T92609 C6-MAR-04 85469868 IC50 = 89.24 nM T92609 CJQ9O7 85469869 IC50 = 49.61 nM T92609 C4HA3I 85469870 IC50 = 227.7 nM T92609 C9NL2S 85469871 IC50 = 96.01 nM T92609 C1J0GW 85469872 IC50 = 551.9 nM T92609 CVM3B2 85469873 IC50 = 384.2 nM T92609 CYI5J6 85469930 IC50 = 34.47 nM T92609 CZI3Y2 85469931 IC50 = 66.23 nM T92609 CAS6Y8 85469932 IC50 = 30.12 nM T92609 C7PXK3 85469933 IC50 = 2.03 nM T92609 C7XI0F 85469934 IC50 = 229.4 nM T92609 CLBA19 86344174 IC50 = 1.9 nM T92609 CL9GY7 90645592 Ki = 1.096 nM T92609 CI49HV 90645593 Ki = 1.479 nM T92609 C41AGZ 90645594 Ki = 7.079 nM T92609 C1L0PW 90645595 Ki = 5.248 nM T92609 C7JL5G 90645596 Ki = 1.096 nM T92609 C89TJI 90645597 Ki = 0.3236 nM T92609 CHBC38 90645598 Ki = 0.9333 nM T92609 C4MLA7 90645599 Ki = 1.622 nM T92609 C0WXR7 90645600 Ki = 6.918 nM T92609 CN8TF6 90645601 Ki = 1.698 nM T92609 CKN56Z 90645602 Ki = 3.89 nM T92609 CYQ3M8 90645603 Ki = 3.388 nM T92609 C45MSD 90645604 Ki = 3.548 nM T92609 C4I6EW 90645605 Ki = 0.912 nM T92609 CH92LD 90645606 Ki = 1 nM T92609 CRX16J 91884611 IC50 = 151 nM T92609 C7YQM3 101333429 Ki = 0.4 nM T92609 CE0ZC6 101876962 Ki = 7 nM T92609 CJ15CM 102012413 Ki = 30 nM T92609 CA43MY 117839022 IC50 = 2.7 nM T92609 C0TMZ8 118167692 IC50 = 8000 nM T92609 C1CP6Z 118567543 Ki = 470 nM T92609 CUV5Y0 118715454 EC50 > 30000 nM T92609 CI7NQ9 118716698 Ki = 8.511 nM T92609 CGO9W4 118716699 Ki = 16.98 nM T92609 CVDI36 118716700 Ki = 6.761 nM T92609 CTX92K 118716702 Ki = 9.772 nM T92609 CG02WP 118716703 Ki = 48.98 nM T92609 CTNL85 118716704 Ki = 6.457 nM T92609 CM1Y8W 118716705 Ki = 17.78 nM T92609 C42MOT 118716706 Ki = 10.72 nM T92609 C78ARU 118716707 Ki = 10.23 nM T92609 CO5TG3 118716708 Ki = 21.38 nM T92609 CNF78L 118716709 Ki = 30.9 nM T92609 C9CB1Q 118716710 Ki = 11.75 nM T92609 C3F6EQ 118716711 Ki = 60.26 nM T92609 C0L6YO 118716712 Ki > 1000 nM T92609 CX2AC4 118716713 Ki = 7.943 nM T92609 CL1EU8 118716714 Ki = 4.571 nM T92609 C0V7GJ 118716715 Ki = 6.457 nM T92609 CRBI65 118716716 Ki = 8.913 nM T92609 C70IPZ 118716717 Ki = 5.248 nM T92609 CBI30N 118716718 Ki = 3.02 nM T92609 C7UBN8 118716719 Ki = 7.943 nM T92609 CV8HA2 118716720 Ki = 18.62 nM T92609 C30ZJB 118716721 Ki = 12.02 nM T92609 C58MND 118716722 Ki = 19.95 nM T92609 CO6T4G 118716723 Ki = 12.59 nM T92609 C8RVX4 118717455 Ki = 134.9 nM T92609 C5IM1N 118717456 Ki = 120 nM T92609 CBCU90 118717457 Ki = 69 nM T92609 CN4LJ2 118717458 Ki = 616.6 nM T92609 CZ35PU 118717459 Ki = 316 nM T92609 C9BP7A 118717460 Ki = 112 nM T92609 CFCM61 118717461 Ki = 257 nM T92609 C8C6ZW 118717462 Ki = 74 nM T92609 CR8Z0F 118718431 Ki = 98 nM T92609 C8Z0PK 118727909 EC50 = 329.1 nM T92609 CT4CW7 118727915 EC50 = 138.2 nM T92609 CFMJ96 119081417 IC50 = 620 nM T92609 CUEG14 122179430 Ki = 0.3 nM T92609 CV51WL 122179431 Ki = 29.9 nM T92609 CUK7B0 122184771 EC50 = 277 nM T92609 CX7U6O 122184772 EC50 = 61 nM T92609 CNT76C 122184833 EC50 > 10000 nM T92609 C8C2KW 122184834 EC50 > 10000 nM T92609 CGNH50 122184835 EC50 = 33 nM T92609 C5PW9Y 123141715 IC50 = 15.4 nM T92609 C03AHG 123183757 IC50 = 4.6 nM T92609 CK4ZO0 123183788 IC50 = 7.6 nM T92609 C17PEO 123204312 IC50 = 21.8 nM T92609 C9W8OX 123311113 IC50 = 38.2 nM T92609 CCK90I 123322716 IC50 = 25.6 nM T92609 C8AKN7 123368349 IC50 = 2.9 nM T92609 C5I2VU 123378354 IC50 = 70.8 nM T92609 C9ZCI2 123387804 IC50 = 20.7 nM T92609 C6LRF9 123393714 IC50 = 324.2 nM T92609 CU7CX9 123415538 IC50 = 2.7 nM T92609 C3HJV5 123437117 IC50 = 8.1 nM T92609 CO3CT2 123472560 IC50 = 2.2 nM T92609 C8RU2P 123475619 IC50 = 3.7 nM T92609 C8XV2H 123562321 IC50 = 0.3 nM T92609 CF2R5U 123576734 IC50 = 57 nM T92609 C1HE3L 123644751 IC50 = 3.2 nM T92609 C9IR4A 123667086 IC50 = 2.7 nM T92609 C3CK5L 123688273 IC50 = 4 nM T92609 CAN97K 123752717 IC50 = 58 nM T92609 C9CO7R 123801568 IC50 = 27.8 nM T92609 CI4TU7 123854385 IC50 = 1.3 nM T92609 C2T0KW 123986550 IC50 = 17.1 nM T92609 C7T0GE 124018870 IC50 = 2.9 nM T92609 CM57GR 126720252 Ki = 1770 nM T92609 CCF0J2 127024958 Ki = 46.7 nM T92609 C82TLX 127024959 Ki = 38.5 nM T92609 C2MWE6 127024960 Ki = 166 nM T92609 C9AQH0 127025258 Ki = 230 nM T92609 CH1CG6 127025275 Ki = 1030 nM T92609 CG3N7S 127025276 Ki = 5 nM T92609 CGO8I5 127025277 Ki = 81 nM T92609 CJZC96 127025278 Ki = 65.5 nM T92609 CQ60XE 127025279 Ki = 418 nM T92609 CTBN56 127026052 Ki = 1258.93 nM T92609 CG8Q4L 127026123 Ki = 29.9 nM T92609 C2YDB4 127027076 Ki = 283 nM T92609 CU59DP 127027077 Ki = 1525 nM T92609 CI94GN 127027078 Ki = 19 nM T92609 C2H6GE 127027079 Ki = 211 nM T92609 C5G4AH 127027080 Ki = 158 nM T92609 C9PNV3 127027384 Ki = 160 nM T92609 CH2BP0 127027974 Ki = 116 nM T92609 CXQ94C 127028034 Ki = 10.3 nM T92609 CZ61LK 127034966 EC50 > 5011.87 nM T92609 CA0SN5 127034967 EC50 > 5011.87 nM T92609 CQ0ZT9 127035062 Ki = 333 nM T92609 CU49VE 127036186 Ki = 1258.93 nM T92609 CG06BD 127036932 Ki = 524.81 nM T92609 CVW71O 127036953 Ki = 630.96 nM T92609 CXR71M 127038002 Ki = 0.4074 nM T92609 CL5N3P 127038713 Ki = 11.22 nM T92609 C89SOL 127040060 Ki = 125.89 nM T92609 CQ3L8Z 127040156 Ki = 30.2 nM T92609 CCH14Q 127041710 IC50 = 36.14 nM T92609 C8A1TO 127043026 IC50 = 453.9 nM T92609 C3GX2A 127044893 IC50 = 14.4 nM T92609 C6P4LV 127044894 IC50 = 4.8 nM T92609 C70SOF 127044906 IC50 = 63.1 nM T92609 C1I6UZ 127044911 IC50 = 4.4 nM T92609 CX9PE0 127044912 IC50 = 2.7 nM T92609 CXKQ86 127044916 IC50 = 8 nM T92609 CL40YC 127045050 IC50 = 8.6 nM T92609 CZS1L6 127049862 IC50 = 35 nM T92609 CZD91J 127049863 IC50 = 120 nM T92609 C6GC0F 129186534 IC50 = 124 nM T92609 C8KM6N 129186554 IC50 = 156 nM T92609 CEZT92 129186564 IC50 = 174 nM T92609 C50GOC 130442480 Ki = 8700 nM T92609 CM04RF 130442572 Ki = 7000 nM T92609 CN2KE8 131978695 IC50 = 124.7 nM T92609 CT81OY 132060776 Ki = 3494 nM T92609 CFXL21 132060812 Ki = 3133 nM T92609 CT58QY 132578518 EC50 = 99.7 nM T92609 C8H7BY 132578519 EC50 = 11.1 nM T92609 CAVB41 132584404 Ki > 10000 nM T92609 C6D1HC 134132279 Ki > 1000 nM T92609 CQ95LB 134133571 Ki > 1995.26 nM T92609 CM4XE8 134133829 Ki = 269.15 nM T92609 CM54ZC 134134752 IC50 = 8669 nM T92609 CBG14F 134136412 EC50 = 34.1 nM T92609 CYXO49 134136428 EC50 = 84.2 nM T92609 CG9J7V 134136763 Ki = 79.43 nM T92609 CKH7W6 134137025 Ki = 57.54 nM T92609 CWQ98O 134137522 IC50 = 2057 nM T92609 C5A6XO 134138438 Ki = 199.53 nM T92609 CP67BZ 134138882 IC50 = 125 nM T92609 CB0S8Y 134139869 Ki = 1.995 nM T92609 C3W5SM 134139893 Ki = 31.62 nM T92609 CHG9Z5 134140686 Ki > 1995.26 nM T92609 CFW7E3 134141385 Ki > 1995.26 nM T92609 C7AQ3Y 134142222 IC50 > 10000 nM T92609 CYW9L4 134142282 IC50 = 17.6 nM T92609 C46ZTY 134143085 Ki > 1000 nM T92609 C3NT1H 134143679 Ki > 1995.26 nM T92609 C2IM4X 134143913 Ki > 1995.26 nM T92609 C7GT5Y 134145079 IC50 = 594 nM T92609 CXN73G 134147055 Ki = 2.754 nM T92609 C1QZ5S 134147190 IC50 = 402.9 nM T92609 CS2OC5 134147929 Ki = 2.951 nM T92609 CYK0E3 134148037 EC50 = 191.6 nM T92609 C94IEA 134148920 EC50 = 148.2 nM T92609 CBU81N 134149168 Ki > 10000 nM T92609 C7HT1Z 134149596 Ki = 0.389 nM T92609 C0CEH2 134149598 IC50 = 253.8 nM T92609 CEU53H 134149777 Ki = 186.21 nM T92609 C91JOU 134150128 IC50 = 2880 nM T92609 C1PQ5T 134150412 Ki > 1995.26 nM T92609 C4BH9V 134150497 Ki = 5.012 nM T92609 CF46WD 134150827 IC50 = 225.3 nM T92609 C3H7KF 134151231 EC50 = 160.7 nM T92609 C9IAC0 134152568 Ki = 2.239 nM T92609 CZ3W6X 134152704 IC50 > 10000 nM T92609 CES7K2 134153419 IC50 > 10000 nM T92609 CDWP64 134153527 Ki > 1000 nM T92609 CJ45MK 134154987 EC50 = 120.6 nM T92609 C4MX2L 134155537 IC50 = 2286 nM T92609 CFW4O8 134156323 EC50 = 140.1 nM T92609 C8KSZ7 134157118 IC50 = 1474 nM T92609 C6S0VM 134157330 Ki = 229.09 nM T92609 CBL29F 134157566 IC50 = 202.3 nM T92609 CEMQ16 134157567 IC50 = 7600 nM T92609 C1GY2T 135156251 EC50 > 10000 nM T92609 CM5F9S 136048765 Ki = 3.6 nM T92609 C25RED 137631359 Ki = 117.49 nM T92609 CST8X9 137637836 Ki = 0.17 nM T92609 C19JKQ 137638321 Ki = 169.82 nM T92609 CA03VC 137639125 Ki = 281.84 nM T92609 CZ4TA9 137640201 Ki = 257.04 nM T92609 CE8N4S 137641762 Ki > 10000 nM T92609 CU1O2P 137642386 Ki = 154.88 nM T92609 CKS5V0 137643541 Ki > 10000 nM T92609 CPCY48 137645406 Ki = 2178 nM T92609 C96EAP 137646245 Ki = 194.98 nM T92609 CPI68E 137646281 Ki = 49 nM T92609 CV29AN 137646446 Ki = 0.18 nM T92609 CW2L7Z 137651819 Ki = 114.82 nM T92609 CR9F3Q 137653203 Ki > 10000 nM T92609 C04XYN 137653567 IC50 = 8.99 nM T92609 CB8C3F 137657762 EC50 = 163 nM T92609 C6QKW5 137659584 Ki = 0.16 nM T92609 CMDV74 144096985 Ki = 50 nM T92609 CN67YQ 144096995 Ki = 150 nM T92609 C91RQY 145949210 Ki = 120.23 nM T92609 CL0XY8 145950240 Ki = 18.2 nM T92609 C45LBY 145951352 Ki = 109.65 nM T92609 CB3O4C 145951457 Ki > 1000 nM T92609 CE3ZM8 145953314 Ki = 5.754 nM T92609 C6VO0S 145955016 Ki > 1000 nM T92609 CT9I0G 145956955 Ki = 0.631 nM T92609 C75KTN 145958538 Ki = 190.55 nM T92609 CX56QA 145960918 Ki = 6.607 nM T92609 CFBX59 145962085 Ki > 1000 nM T92609 C2FNR9 145962342 Ki = 1.862 nM T92609 CE9I6G 145962368 Ki = 22.39 nM T92609 C0G7JA 145962478 Ki = 7.079 nM T92609 C3DGE5 145962817 Ki = 223.87 nM T92609 C2HL4E 145962945 Ki = 16.98 nM T92609 C7BC0I 145963755 Ki = 33.11 nM T92609 C64TUP 145963761 Ki = 1800 nM T92609 CQU59F 145963832 Ki > 270 nM T92609 CEN94V 145963961 IC50 = 71 nM T92609 C1B8QW 145964299 IC50 = 11 nM T92609 C95NZO 145964427 Ki = 14 nM T92609 C6T4RY 145964846 Ki = 93 nM T92609 C9D8IB 145965203 Ki = 11 nM T92609 CZ86PI 145965488 Ki = 1200 nM T92609 C0TU9I 145965623 Ki = 220 nM T92609 CLM10C 145966333 IC50 = 164 nM T92609 CZSN84 145967270 Ki > 270 nM T92609 CBPU13 145968055 IC50 = 1073.85 nM T92609 CTJ0X5 145968736 IC50 = 502.12 nM T92609 CTP81Y 145968741 IC50 = 57.58 nM T92609 C9M7ZG 145969396 Ki > 270 nM T92609 CT9FQ7 145969986 IC50 = 567.63 nM T92609 CDLX87 145970204 IC50 = 1212.48 nM T92609 C7IGH9 145970995 Ki = 350 nM T92609 CEOY46 145973577 Ki = 36 nM T92609 CQIB05 145975238 Ki = 130 nM T92609 CF8ET9 145975365 Ki > 270 nM T92609 CL7EX5 145975776 Ki = 772 nM T92609 C8XFM7 145976120 Ki = 2117 nM T92609 C34XME 145976696 Ki = 15 nM T92609 C0W3YR 145977627 Ki > 270 nM T92609 C1DW4U 145983928 IC50 = 178 nM T92609 CI0PA9 145987771 Ki = 28 nM T92609 CMJ46R 145990794 IC50 = 124 nM T92609 C9PS8N 145993117 IC50 = 376 nM T92609 C0Z6YX 145993493 IC50 = 375 nM T92609 CC2G1V 146025727 Ki = 2900 nM T92609 C6P3SR 153287553 Ki > 10000 nM T92609 CV9G7Z 153287572 Ki > 10000 nM T92609 CO85KL 153287574 Ki = 1584.89 nM T92609 C7N0VH 155512508 Ki > 1000 nM T92609 C7W1OH 155513940 Ki = 83.18 nM T92609 CV8F7A 155515301 Ki = 354.81 nM T92609 CUM2N4 155515982 Ki = 1.7 nM T92609 CT4U8D 155517137 Ki > 1000 nM T92609 CAV5Y1 155519565 Ki > 1000 nM T92609 CUSA24 155519891 Ki > 10000 nM T92609 CL07FB 155521817 Ki > 1000 nM T92609 CXEB36 155523275 Ki > 1000 nM T92609 CYZ60F 155524736 Ki > 1000 nM T92609 CD5BI1 155525649 Ki = 120.23 nM T92609 C8GC1P 155526628 Ki = 7.244 nM T92609 CIO6V1 155528183 Ki > 1000 nM T92609 C7FR8Y 155529117 Ki = 426.58 nM T92609 CF2DM6 155529314 Ki = 16.98 nM T92609 C3ZL2V 155531279 Ki > 1000 nM T92609 C3R4YM 155532148 Ki = 2.63 nM T92609 C3MXL6 155532834 Ki = 24.55 nM T92609 CTU64O 155533099 Ki = 44.67 nM T92609 CU3YE7 155534933 Ki > 1000 nM T92609 CB79ZW 155536080 Ki > 10000 nM T92609 CQG68A 155536202 Ki = 169.82 nM T92609 CFH7K5 155542074 Ki = 58.88 nM T92609 C91VXF 155544397 Ki > 1000 nM T92609 CR54LA 155544513 Ki = 977.24 nM T92609 CXH9A8 155549493 Ki > 1000 nM T92609 CX8JA1 155552185 Ki = 1.6 nM T92609 C9XQ8H 155552820 Ki = 288.4 nM T92609 C4LOH3 155555858 Ki = 60.26 nM T92609 C0CV6O 155557695 Ki = 141.25 nM T92609 C3UCM2 155557792 Ki > 1000 nM T92609 C20QMI 155558704 Ki > 1000 nM T92609 CE0HN5 155559841 Ki > 1000 nM T92609 C8ZKT3 155562124 Ki = 38.9 nM T92609 C71MOD 155563001 Ki = 30.9 nM T92609 C3DK0P 155565218 Ki = 89.13 nM T92609 CVU9O2 155565448 Ki = 50.12 nM T92609 C19PZX 155565707 Ki > 1000 nM T92609 CRX52O 155567200 Ki = 33.88 nM T92609 C3N9VU 10251906 Ki > 500 nM T92609 CB2VD8 44241743 Ki = 73 nM T92609 D00GEE 92766 Ki = 29 nM T92609 D01BJZ 9817640 Ki = 3.981 nM T92609 D01KAX 135453290 Ki > 30000 nM T92609 D02NNS 9845181 Ki = 290 nM T92609 D02YSX 197033 Ki = 60.26 nM T92609 D05EQG 5265 Ki = 7.9 nM T92609 D05GDP 599482 Ki > 10000 nM T92609 D05ZUX 44207909 Ki = 260 nM T92609 D06ABL 9891980 Ki = 10.34 nM T92609 D06QKW 2765 EC50 = 12.59 nM T92609 D06UBB 123981 Ki = 449 nM T92609 D07OAF 4038180 EC50 = 9.3 nM T92609 D07QCC 10946567 Ki = 58 nM T92609 D08HOJ 34677 EC50 > 30000 nM T92609 D08XTL 9866614 Ki = 0.65 nM T92609 D09CUJ 1862 Ki = 1500 nM T92609 D09RPR 16737207 Ki > 10000 nM T92609 D09WIL 10028436 Ki = 218.78 nM T92609 D09ZUW 6603904 Ki = 420 nM T92609 D0A0JU 6603710 Ki = 490 nM T92609 D0C7SE 16756754 Ki = 180 nM T92609 D0D8GV 9830741 Ki = 0.17 nM T92609 D0DP8I 132266 Ki = 5.495 nM T92609 D0EO4F 9891167 Ki = 4.17 nM T92609 D0H3CW 9839317 Ki = 3300 nM T92609 D0HH3R 11698643 Ki = 78 nM T92609 D0L5MW 181743 Ki = 2 nM T92609 D0M5ZE 5311416 Ki = 316.23 nM T92609 D0N0SN 44390756 Ki = 59 nM T92609 D0N7UE 10198248 Ki = 18197.01 nM T92609 D0O3GF 1220 Ki = 151.36 nM T92609 D0O6MG 3567002 Ki = 0.25 nM T92609 D0P4KF 44269078 Ki = 91 nM T92609 D0PN9R 16655023 Ki = 125 nM T92609 D0Q4PY 9888164 Ki = 18 nM T92609 D0Q7ZR 9890547 Ki = 2.6 nM T92609 D0R4MH 22629308 Ki = 41 nM T92609 D0T2RY 9948320 Ki = 18 nM T92609 D0V6DJ 5640 Ki = 0.631 nM T92609 D0XL9J 44390740 Ki = 5 nM T92609 D0Z7EA 643606 Ki = 4400 nM T92609 D0Z8OD 9887378 Ki = 8.7 nM T76910 D02ZQS 16095342 IC50 = 1260 nM T76910 D06DMQ 59472121 Ki = 33 nM T76910 D08HOM 46207586 IC50 > 10000 nM T76910 D0CY1B 6420138 Ki > 10000 nM T76910 D0E3TC 44259 IC50 = 2.4 nM T76910 D0Z1DH 10029385 IC50 = 1.02 nM T76910 D03BNU 59604787 IC50 > 10000 nM T76910 D00OWF 5280953 IC50 > 10000 nM T76910 D0A3MV 448014 IC50 = 70000 nM T76910 D0NS6I 10037501 IC50 = 7700 nM T76910 D0Q3VZ 135398522 IC50 = 210 nM T76910 D0WX0K 71680628 IC50 = 40 nM T76910 D0YK9D 9956119 IC50 = 7.8 nM T76910 C6WUY3 3513 IC50 = 26 nM T76910 C0FK8L 726568 IC50 = 145 nM T76910 CXO42B 805390 IC50 = 2244 nM T76910 C53QBZ 837609 IC50 = 904 nM T76910 CQ1YV2 904180 IC50 = 609 nM T76910 C7XUM0 1026218 IC50 = 10160 nM T76910 C1Q4XB 1051604 IC50 = 440 nM T76910 CA0QI6 1227680 IC50 = 2804 nM T76910 CI40FJ 1232232 IC50 = 16830 nM T76910 CA3GF2 1467927 IC50 = 7379 nM T76910 CX23OE 1729742 IC50 > 100000 nM T76910 CJ57GZ 1842529 IC50 = 557 nM T76910 C29TYV 2673354 IC50 = 15 nM T76910 C3ZI1K 2764173 IC50 > 5000 nM T76910 C86LNP 2779952 IC50 > 100000 nM T76910 C1KPM5 3123256 IC50 = 12980 nM T76910 CO53NJ 5194305 IC50 = 4600 nM T76910 CK7Y6A 5718019 IC50 = 412 nM T76910 CW1EK3 5881165 IC50 = 309 nM T76910 C7EMW0 5919090 IC50 = 33 nM T76910 CB2TY1 5998116 IC50 = 370 nM T76910 CEZP52 6263849 IC50 = 250 nM T76910 CH13FR 6538884 IC50 = 530 nM T76910 CV1EC6 6539452 IC50 = 216000 nM T76910 C0MW6H 6539453 IC50 = 216000 nM T76910 C95UNH 6539454 IC50 = 141000 nM T76910 CHQB47 6539455 IC50 = 514000 nM T76910 CK0QF7 6539456 IC50 = 390000 nM T76910 CC2N8D 6539457 IC50 = 301000 nM T76910 CO5ZI9 6539458 IC50 = 195000 nM T76910 CUQ6F3 6539459 IC50 = 114000 nM T76910 CD94GZ 6539460 IC50 = 104000 nM T76910 CXI9R2 6539461 IC50 = 257000 nM T76910 COG8F9 6539462 IC50 = 70000 nM T76910 CSN2M8 6539463 IC50 = 447000 nM T76910 C7G9QY 6539464 IC50 = 156 nM T76910 C09GEI 6539465 IC50 = 704000 nM T76910 C4MA9R 6539466 IC50 = 374000 nM T76910 C3B1MV 6539467 IC50 = 259000 nM T76910 CZC31W 6539468 IC50 = 251000 nM T76910 CC17FL 6539469 IC50 = 1478000 nM T76910 CT8Z5A 6539470 IC50 = 472000 nM T76910 CQ8P2W 6539471 IC50 = 236000 nM T76910 C0CPN8 6539472 IC50 = 407000 nM T76910 C7OFY0 6539473 IC50 = 481000 nM T76910 CXQB76 6539474 IC50 = 123000 nM T76910 CSYM79 6539475 IC50 = 317000 nM T76910 CX1PB2 6539476 IC50 = 152000 nM T76910 CD0MK5 6539477 IC50 = 139000 nM T76910 C0V8PK 6539478 IC50 = 94000 nM T76910 CW1FA4 6539479 IC50 = 59000 nM T76910 CQT3S5 6539480 IC50 = 173000 nM T76910 CMHO38 6539481 IC50 = 149000 nM T76910 CRB06P 6539482 IC50 = 93000 nM T76910 C0QV9A 6539483 IC50 = 82000 nM T76910 CB1I5W 6539484 IC50 = 52000 nM T76910 CO4EP0 6539485 IC50 = 58000 nM T76910 C15YWK 6539486 IC50 = 142000 nM T76910 CB01VH 6539487 IC50 = 20000 nM T76910 CBZ2U6 6539488 IC50 = 91000 nM T76910 C0CA1Y 6539489 IC50 = 83000 nM T76910 C3ZF8P 6539490 IC50 = 71000 nM T76910 CEI56T 6539491 IC50 = 291000 nM T76910 CR3A6L 6539492 IC50 = 136000 nM T76910 CT2H9L 6539493 IC50 = 134000 nM T76910 C9LYZ2 6539494 IC50 = 195000 nM T76910 C0ZDY3 6539495 IC50 = 79000 nM T76910 CR72NT 6539496 IC50 = 186000 nM T76910 C6DKW8 6539497 IC50 = 214000 nM T76910 CD0T4H 6539498 IC50 = 143000 nM T76910 CXS64M 6539499 IC50 = 74000 nM T76910 CI2AZ0 6539500 IC50 = 28 nM T76910 C5YWB1 6539501 IC50 = 85000 nM T76910 CX9V7E 6539502 IC50 = 109000 nM T76910 CUWN19 6539503 IC50 = 404000 nM T76910 C0P3JF 6539504 IC50 = 161000 nM T76910 CG8Q3U 6539505 IC50 = 110000 nM T76910 CM58CR 6539506 IC50 = 532000 nM T76910 CN4JS2 6539507 IC50 = 203000 nM T76910 CNE79Y 6539508 IC50 = 152000 nM T76910 C3YRL2 6539509 IC50 = 529000 nM T76910 CY5NZ6 6539510 IC50 = 243000 nM T76910 CP86TH 6539511 IC50 = 392000 nM T76910 C8D5RK 6539512 IC50 = 2613000 nM T76910 CS1LT5 6539513 IC50 > 4500000 nM T76910 C5T8YX 6539514 IC50 = 1398000 nM T76910 C1K8EO 6539515 IC50 = 2285000 nM T76910 CILQ58 6539516 IC50 = 337000 nM T76910 CA9KF0 6539517 IC50 = 187 nM T76910 CLV36F 6539518 IC50 = 131000 nM T76910 C37DQI 6539519 IC50 = 460000 nM T76910 CX7A4E 6539520 IC50 = 161000 nM T76910 CD4A1X 6539521 IC50 = 1412000 nM T76910 CXS23C 6539522 IC50 = 694000 nM T76910 C6R3GO 6539523 IC50 > 5000 nM T76910 CIN73F 6539524 IC50 > 5000 nM T76910 C6IH1C 6539525 IC50 > 3000 nM T76910 CF3S6U 6539526 IC50 = 7 nM T76910 CE75FM 6539527 IC50 = 4 nM T76910 CG8ZC5 6539528 IC50 = 430 nM T76910 CVE25D 6539529 IC50 = 1260 nM T76910 CR7JG1 6539530 IC50 > 5000 nM T76910 C5J1RN 6539531 IC50 > 5000 nM T76910 C7RA9C 6539532 IC50 > 5000 nM T76910 C0GI9Y 6539533 IC50 = 291 nM T76910 CL54CB 6539534 IC50 = 43 nM T76910 C8ZTV0 6539535 IC50 = 56 nM T76910 CETM71 6539536 IC50 = 19 nM T76910 CKM15E 6539537 IC50 = 5 nM T76910 CFS2R3 6539538 IC50 = 2810 nM T76910 C31TYK 6539539 IC50 = 3572 nM T76910 C0MG7X 6539540 IC50 = 356 nM T76910 CP7SM9 6539541 IC50 = 2345 nM T76910 CX90YS 6539542 IC50 = 18 nM T76910 C63YHD 6539543 IC50 = 20 nM T76910 C8BD2P 6539544 IC50 = 7 nM T76910 CJI31S 6539545 IC50 = 27 nM T76910 CX6M9C 6539546 IC50 = 11 nM T76910 C3JBE0 6539547 IC50 = 443 nM T76910 C53JWE 6539548 IC50 = 851 nM T76910 C87EVK 6539549 IC50 = 169 nM T76910 CVGH07 6539550 IC50 = 241 nM T76910 CQ74FL 6539551 IC50 = 99 nM T76910 C5M3BE 6539552 IC50 = 2697 nM T76910 C9D1ME 6539553 IC50 = 691 nM T76910 CU61ZB 6539554 IC50 = 22 nM T76910 CL2RW0 6539555 IC50 = 11 nM T76910 C5SGK0 6539556 IC50 = 7 nM T76910 CXV5C7 6539557 IC50 = 5 nM T76910 C7L2OQ 6539558 IC50 = 9 nM T76910 CTU82J 6539559 IC50 = 5 nM T76910 C9V5PK 6539560 IC50 = 5 nM T76910 CL20EZ 6539565 IC50 = 425 nM T76910 CMN15O 6539567 IC50 > 5000 nM T76910 CP7J3S 6539569 IC50 = 12 nM T76910 CS6T9C 6539570 IC50 = 125 nM T76910 C8B5SQ 6539572 IC50 = 1593 nM T76910 CC12VG 6539577 IC50 = 415 nM T76910 C7C9BO 6539578 IC50 = 75 nM T76910 CIT1W5 6539579 IC50 = 234 nM T76910 CVSZ60 6539580 IC50 = 87 nM T76910 C0V5BI 6539581 IC50 = 383 nM T76910 CX9V6S 6539585 IC50 = 21 nM T76910 CCXU69 6539586 IC50 = 215 nM T76910 CQTU34 6539587 IC50 = 329 nM T76910 COI57D 6539588 IC50 = 39 nM T76910 CQ97IV 6539591 IC50 = 7 nM T76910 C70OTV 6539592 IC50 = 141 nM T76910 CAI54V 6539593 IC50 = 498 nM T76910 C9ABL1 6539595 IC50 = 42 nM T76910 C87GNI 6539596 IC50 > 1000 nM T76910 CGO8A0 6539597 IC50 > 1000 nM T76910 C4TJI2 6539598 IC50 = 481 nM T76910 CHWL84 6539599 IC50 > 1000 nM T76910 C6P4BO 6539600 IC50 > 1000 nM T76910 CG1C4I 6539601 IC50 > 1000 nM T76910 CHP97J 6539602 IC50 > 1000 nM T76910 C79LMV 6539603 IC50 > 1000 nM T76910 CDS2B8 6539604 IC50 > 1000 nM T76910 CWJ6C1 6539605 IC50 > 1000 nM T76910 CNV39L 6539606 IC50 = 828 nM T76910 CH54ZS 6539607 IC50 > 1000 nM T76910 C14VJA 6539608 IC50 = 320 nM T76910 C1M3ZI 6539609 IC50 = 50 nM T76910 C7U2TC 6539610 IC50 = 35 nM T76910 C5XBK1 6539611 IC50 = 7 nM T76910 CNE0Y5 6539612 IC50 = 99 nM T76910 CK3W6M 6539613 IC50 = 16 nM T76910 CJV73P 6539614 IC50 = 18 nM T76910 C1PVJ8 6539615 IC50 = 14 nM T76910 CY20RA 7458031 IC50 = 9 nM T76910 C2B4OG 7857292 IC50 = 15 nM T76910 CQ57EC 9548013 IC50 > 100000 nM T76910 CD5H7P 9607118 IC50 = 11210 nM T76910 C2W3AV 9995236 IC50 = 900 nM T76910 CBOP58 11293798 Ki > 10000 nM T76910 C26BZX 11362471 Ki > 10000 nM T76910 CWXB93 11397177 Ki > 10000 nM T76910 CTG83F 11539329 Ki > 8900 nM T76910 CMIL86 11590363 Ki > 8900 nM T76910 CU7WH8 11601694 IC50 = 330 nM T76910 C9T6SC 11640926 Ki > 8900 nM T76910 CTI2R7 11856271 IC50 = 123 nM T76910 C64JCR 11856273 IC50 = 61 nM T76910 CV9T5S 11856528 IC50 = 1499 nM T76910 COT84C 11856529 IC50 = 91 nM T76910 CD9A7C 11856530 IC50 = 133 nM T76910 CHJ01P 13303387 IC50 > 10000 nM T76910 C5YF0D 13303393 IC50 > 10000 nM T76910 CFPW41 16007116 Ki > 8900 nM T76910 C7Z4LV 16095343 IC50 = 9100 nM T76910 C5VPH9 16129448 IC50 > 10000 nM T76910 C9FMS4 16374676 IC50 = 3206 nM T76910 CB7U1R 17408143 IC50 = 451 nM T76910 CC2UB6 21214332 IC50 = 710 nM T76910 CY6CQ1 21214334 IC50 = 159 nM T76910 C8AMQ9 23641602 IC50 = 22 nM T76910 CFMQ08 24370907 IC50 = 52 nM T76910 C7YG1N 24759534 IC50 = 360 nM T76910 CV79PK 24984058 IC50 = 990 nM T76910 CX1HL8 25032704 Ki = 1110 nM T76910 C0OW7X 25167905 IC50 = 4.5 nM T76910 C8KH9R 29998963 IC50 = 6150 nM T76910 C2U0NP 30291209 IC50 < 5 nM T76910 C7S6OT 30291292 IC50 = 19 nM T76910 C32ZDN 44307910 IC50 = 6.2 nM T76910 CS2G7K 44448292 IC50 = 9 nM T76910 C4E5DN 44448294 IC50 = 13 nM T76910 CU06RO 44448295 IC50 = 74 nM T76910 CFW9Q8 44448296 IC50 = 123 nM T76910 CD3N2S 44448318 IC50 = 20 nM T76910 C54FTS 44448319 IC50 = 172 nM T76910 C4C2EM 44448320 IC50 = 32 nM T76910 C7JV9D 44448340 IC50 = 6700 nM T76910 CAK9P5 44448341 IC50 = 1900 nM T76910 C2YK7C 44448342 IC50 = 350 nM T76910 C7Y1SX 44448360 IC50 = 1020 nM T76910 CSE08W 44448362 IC50 = 750 nM T76910 CLCO97 44448363 IC50 = 3760 nM T76910 CNGP68 44448395 IC50 = 1870 nM T76910 CK6WJ8 44448397 IC50 = 270 nM T76910 CP07GH 44448693 IC50 = 444 nM T76910 CT24RL 44448694 IC50 = 38 nM T76910 CX0QU1 44448695 IC50 = 96 nM T76910 C3ZHT1 44448715 IC50 = 66 nM T76910 C08EFA 44448716 IC50 = 80 nM T76910 CK0S7D 44448735 IC50 = 34 nM T76910 CVA38F 44448737 IC50 = 204 nM T76910 C79YQL 44448738 IC50 = 23 nM T76910 CYH6P3 44520205 IC50 = 5340 nM T76910 C4WRN5 44541014 IC50 = 10.6 nM T76910 C3VRO9 44557921 IC50 > 10000 nM T76910 CY3HW5 46224684 IC50 = 170 nM T76910 CLS29B 46872626 IC50 > 10000 nM T76910 C2O8RZ 46886323 IC50 > 1000 nM T76910 CB0S2P 49842666 IC50 > 100000 nM T76910 CAI20B 49842778 IC50 > 100000 nM T76910 CU90AO 50942121 Ki = 9 nM T76910 C6M9TQ 51039273 IC50 > 100000 nM T76910 CS7Q3D 51347384 IC50 > 100000 nM T76910 C16UXT 51347682 IC50 > 100000 nM T76910 CJU19H 51347839 IC50 > 100000 nM T76910 CE9TJ5 51347987 IC50 > 25000 nM T76910 C71OXL 53388145 IC50 = 130000 nM T76910 CDL28G 53388146 IC50 = 370000 nM T76910 C2G3AY 54726684 IC50 = 1621.81 nM T76910 CIM94L 56668847 IC50 = 220000 nM T76910 C8PK0W 56675716 IC50 = 1120000 nM T76910 C2VPR0 57397894 IC50 = 600 nM T76910 CFZ40T 57522594 IC50 = 107 nM T76910 CEW5L7 57522817 IC50 = 2 nM T76910 C4SEH5 57522818 IC50 = 6 nM T76910 CF8IP6 57522819 IC50 < 5 nM T76910 CJ56CE 57522820 IC50 = 2 nM T76910 C3XI2P 57523093 IC50 = 54 nM T76910 CUH3B5 57523094 IC50 = 195 nM T76910 C3QF2X 57523095 IC50 = 15 nM T76910 CXJ63M 59603829 IC50 = 130 nM T76910 CQEU96 59603842 IC50 = 42 nM T76910 C37NKO 67129970 IC50 = 9360 nM T76910 CK80LJ 67130050 IC50 > 10000 nM T76910 CV63UL 67240318 IC50 > 5000 nM T76910 C7GRV2 68755406 IC50 > 10000 nM T76910 C5DGR9 69036886 IC50 = 3308 nM T76910 CNKB34 70682366 IC50 = 45 nM T76910 C0RT2G 70690776 IC50 = 95 nM T76910 C2XV4Q 70694953 IC50 = 12 nM T76910 CL1HY5 71212233 IC50 = 195 nM T76910 CKX52R 71212291 IC50 = 9 nM T76910 C0T2VB 71212317 IC50 = 5 nM T76910 C5B8NS 71212337 IC50 = 15 nM T76910 CSN04E 71212395 IC50 = 19 nM T76910 C1OCW0 71212403 IC50 = 240 nM T76910 CBX2I4 71212419 IC50 = 51 nM T76910 CLS4R3 71212434 IC50 = 77 nM T76910 CTF8M7 71212446 IC50 = 5 nM T76910 C2Z8CX 71212514 IC50 = 46 nM T76910 CBT7L3 71212517 IC50 = 35 nM T76910 CKT60L 71455860 Ki = 21 nM T76910 CY6WI2 71458575 IC50 = 260 nM T76910 CHY91V 71578307 IC50 = 4 nM T76910 C0W2KX 71578373 IC50 = 3 nM T76910 C6TX9R 71578374 IC50 = 4 nM T76910 C2D1RN 71578375 IC50 = 15 nM T76910 C73MEW 71578445 IC50 = 7 nM T76910 C5NH3V 71578446 IC50 = 51 nM T76910 CC65WU 71578447 IC50 = 27 nM T76910 CIP6Q2 71578520 IC50 = 324 nM T76910 CPJ19D 71578658 IC50 = 20 nM T76910 C5W0GC 71578744 IC50 = 17 nM T76910 CLZ59B 71578745 IC50 = 2 nM T76910 C4B5RW 72725141 IC50 = 884 nM T76910 CRE2U3 77050682 IC50 = 462 nM T76910 C1HW4B 89735655 IC50 = 110 nM T76910 CK7D6O 118879529 IC50 = 691 nM T76910 C32YBQ 122194770 IC50 = 42 nM T76910 C8S0OH 135416016 IC50 = 24 nM T76910 C3YPB0 135416046 IC50 = 4 nM T76910 C52RQG 135435008 IC50 = 8 nM T76910 CBN98A 135435009 IC50 = 8 nM T76910 CN6HJ9 135435010 IC50 = 36 nM T76910 CPFI68 135435011 IC50 = 0.8 nM T76910 C97ABO 135435012 IC50 = 1 nM T76910 CPXC89 135435013 IC50 = 6 nM T76910 CIX53V 135435014 IC50 = 12 nM T76910 CNM94K 135435015 IC50 = 1 nM T76910 CS14KX 135435016 IC50 = 5 nM T76910 C2ICP3 135435017 IC50 = 7 nM T76910 C6AZ2R 135435018 IC50 = 15 nM T76910 C09BEG 135486057 IC50 > 10000 nM T76910 CG9R0V 135741827 IC50 > 10000 nM T76910 C5RI6D 136224254 IC50 > 10000 nM T76910 CT9VC6 136224366 IC50 > 10000 nM T76910 CF6B3S 136224367 IC50 > 10000 nM T76910 C6S1GT 136245126 IC50 > 10000 nM T76910 CS6K0B 136245127 IC50 > 10000 nM T76910 CA5KP8 136245128 IC50 > 10000 nM T76910 C8UQ7C 136264319 IC50 > 10000 nM T76910 CNE6I8 136264499 IC50 > 10000 nM T76910 C7EAJ9 136980453 IC50 = 66 nM T76910 C6R2PY 137630916 IC50 = 1340 nM T76910 CI1E8V 137634241 IC50 > 10000 nM T76910 CDA2N6 137644922 IC50 = 37 nM T76910 CA3G0W 140534484 IC50 = 207 nM T76910 CL48DN 145951168 IC50 = 4 nM T76910 C4K8TH 154777683 IC50 = 282 nM T76910 CUP08F 154778142 IC50 = 242 nM T76910 CRAD72 154778144 IC50 = 1879 nM T76910 CUH9P6 155077159 IC50 = 301 nM T76910 C2MD1Q 155513187 IC50 > 10000 nM T76910 C76ZQG 155524866 IC50 = 49 nM T76910 C5H1UB 155526385 IC50 = 2676 nM T76910 C3ZHC0 155537470 IC50 = 300 nM T76910 COE67I 155538620 IC50 = 428 nM T76910 CDM03I 155541927 IC50 = 301 nM T76910 C3J8SM 155542090 IC50 = 2046 nM T76910 COG6I5 155548241 IC50 = 227 nM T76910 C9C4XO 155553435 IC50 = 853 nM T76910 C48FUJ 155558812 IC50 = 162 nM T76910 CGX17T 155567824 IC50 = 1337 nM T76910 CP06DW 155569342 IC50 = 300 nM T76910 D00ERW 44444843 Ki = 911 nM T76910 D00HVA 11624601 Ki > 8900 nM T76910 D01MEP 6539732 IC50 = 390 nM T76910 D01OJG 6539451 IC50 = 529000 nM T76910 D02OPH 448008 IC50 = 76000 nM T76910 D02XHC 448912 IC50 = 500 nM T76910 D04ZWF 53396311 IC50 = 7 nM T76910 D0A1YQ 176158 IC50 = 34 nM T76910 D0H3EV 5005498 IC50 = 4 nM T76910 D0N4WB 4210951 IC50 = 104 nM T76910 D0Q3KS 9957049 IC50 = 0.65 nM T76910 D0Q3NG 11715520 Ki > 8900 nM T76910 D0Q4QF 6509753 IC50 = 25000 nM T76910 D0S7IE 11658882 Ki > 8900 nM T09909 D06UDG 60846 Ki > 10000 nM T09909 D0D5SQ 2541 Ki > 10000 nM T09909 D0G6SE 172198 Ki = 0.2 nM T09909 D0K0AT 6324663 Ki = 0.15 nM T09909 D0N6RF 65999 IC50 = 0.33 nM T09909 D05FUU 9802561 IC50 > 10000 nM T09909 D0O0JP 9937291 IC50 = 0.58 nM T09909 D00UBK 9851889 IC50 = 0.7 nM T09909 D07LEW 131590 Ki = 480 nM T09909 D0A8HL 3081289 IC50 > 1000 nM T09909 D0F5VB 5311345 IC50 = 6.9 nM T09909 D0GS7N 183134 IC50 = 0.2 nM T09909 D0N5CT 132404 Ki = 730 nM T09909 CTCP47 130762 IC50 = 200 nM T09909 C08QYK 5311348 IC50 = 66 nM T09909 C7SLB9 5748345 Ki = 0.11 nM T09909 CTM56O 9806878 Ki = 4 nM T09909 CZI91W 9807029 IC50 = 775 nM T09909 CH2FD7 9809280 IC50 = 920 nM T09909 C35FCP 9810305 IC50 = 18 nM T09909 C32SAX 9846535 IC50 = 275 nM T09909 C1I6GK 9850811 IC50 = 200 nM T09909 CIWU91 9850834 Ki = 1.5 nM T09909 CV07NF 9851082 IC50 = 1 nM T09909 C2C4OM 9852384 IC50 = 101 nM T09909 CRP84D 9853391 IC50 = 0.12 nM T09909 C9HI0W 9870559 IC50 = 1.1 nM T09909 C6SHG0 9874508 IC50 = 6.2 nM T09909 CK1N5Q 9892451 IC50 = 0.84 nM T09909 CV8A6J 9895212 IC50 = 18 nM T09909 C2M4BW 9895984 IC50 = 60 nM T09909 CI4A8R 9915892 IC50 = 60 nM T09909 CY9N3R 9918412 IC50 = 0.9 nM T09909 C65CYH 9940350 IC50 = 0.69 nM T09909 CG0ET4 9987414 IC50 = 2.9 nM T09909 C8J4GU 10005139 IC50 = 10 nM T09909 C59NJL 10009984 IC50 = 2.7 nM T09909 CE5H3C 10010071 IC50 = 1.2 nM T09909 CEI76X 10010164 IC50 = 3.7 nM T09909 CCS31D 10032820 IC50 = 3.1 nM T09909 CE9XN3 10032851 IC50 = 2.3 nM T09909 CY62AG 10032877 IC50 = 2.6 nM T09909 CT6M8J 10032988 IC50 = 3.8 nM T09909 CJ3D0B 10033136 IC50 = 1.5 nM T09909 CQ1OW7 10034086 Ki = 2.1 nM T09909 CJI2W4 10049400 IC50 = 22 nM T09909 CQUS95 10053595 IC50 = 50 nM T09909 C35BSX 10057017 Ki = 3 nM T09909 C8CDV2 10078320 IC50 = 2.1 nM T09909 CRS30P 10078475 IC50 = 10 nM T09909 CCM3D8 10078554 IC50 = 1.1 nM T09909 C3KX6E 10078780 IC50 = 2.2 nM T09909 C6YFD0 10078800 IC50 = 17 nM T09909 CNQ97X 10079601 Ki = 0.14 nM T09909 CDX49R 10092454 IC50 = 20 nM T09909 CS73XM 10100951 IC50 = 5.8 nM T09909 CM9N8U 10101351 IC50 = 1.4 nM T09909 CS7A5F 10101606 IC50 = 0.64 nM T09909 C3F0TU 10101608 IC50 = 3.7 nM T09909 CFN78G 10101690 IC50 = 6.3 nM T09909 C0TE1A 10116410 Ki = 37 nM T09909 CNIV38 10140382 Ki = 63 nM T09909 C8WK1N 10140383 Ki = 5 nM T09909 CHI2C9 10160913 Ki = 10 nM T09909 CHZ35S 10161763 Ki = 75 nM T09909 CSZ41X 10163396 Ki = 1 nM T09909 CB4CR7 10182998 Ki = 79 nM T09909 C4XFD9 10196520 Ki = 3.2 nM T09909 CI2U7M 10205901 Ki = 86 nM T09909 C8C1LD 10227337 Ki = 13 nM T09909 C4ZSK2 10259265 IC50 = 0.82 nM T09909 CU58CL 10259447 IC50 = 2 nM T09909 CEYO10 10259468 IC50 = 2.2 nM T09909 CUA9G7 10259525 IC50 = 5.3 nM T09909 CI0WR6 10259841 IC50 = 2 nM T09909 C82KRW 10272250 Ki > 10000 nM T09909 C59JVW 10276878 Ki = 5 nM T09909 C9RQA4 10277322 Ki = 31 nM T09909 CVPD28 10289461 Ki = 7.1 nM T09909 CVB1D4 10300357 Ki = 76 nM T09909 CJ9H8M 10327309 IC50 = 4.6 nM T09909 CNZ05L 10327728 IC50 = 4.1 nM T09909 CUQ92S 10344854 IC50 = 50 nM T09909 CLIH83 10349897 IC50 = 2.1 nM T09909 CX1A2T 10350123 IC50 = 3.5 nM T09909 CK24ZW 10372451 IC50 = 3.7 nM T09909 C8PUW5 10372550 IC50 = 7.5 nM T09909 CAU4G3 10372659 IC50 = 3.1 nM T09909 CWAP07 10372810 IC50 = 2.4 nM T09909 CDJ5M3 10373120 IC50 = 5.1 nM T09909 C8EBV1 10391038 IC50 = 5870 nM T09909 C5KEW8 10394727 IC50 = 20 nM T09909 CA07JQ 10394859 IC50 = 1.5 nM T09909 C2WXC5 10395076 IC50 = 1.8 nM T09909 CQB57G 10395335 IC50 = 1.3 nM T09909 C7DL0F 10396262 Ki = 463.7 nM T09909 C42BDV 10414470 IC50 = 789 nM T09909 CB0ZK1 10417195 IC50 = 2.6 nM T09909 C8QY7E 10417321 IC50 = 1.7 nM T09909 CJHU16 10429298 IC50 = 200 nM T09909 C6FSG7 10439715 IC50 = 3.4 nM T09909 C41IQS 10439819 IC50 = 4.1 nM T09909 CO1V5L 10439837 IC50 = 4.3 nM T09909 C9GM1L 10439858 IC50 = 8.2 nM T09909 CG1Q7I 10440144 IC50 = 3.6 nM T09909 CVO28P 10462053 IC50 = 0.9 nM T09909 CT61DH 10462573 IC50 = 3.6 nM T09909 C8PCF5 10462598 IC50 = 4.3 nM T09909 CV93HT 10462683 IC50 = 2.6 nM T09909 CCG2B9 10462933 IC50 = 6.1 nM T09909 CA4K0Y 10463891 Ki = 0.8 nM T09909 CW90RU 10742620 Ki = 480 nM T09909 C0HCU1 11157870 Ki > 10000 nM T09909 CV2MF5 11180576 Ki = 400 nM T09909 CE6W1I 11181498 Ki = 4.6 nM T09909 CCW8H2 11202336 Ki > 10000 nM T09909 C3ISB8 11216369 Ki = 33 nM T09909 CE0S5Y 11239632 Ki = 8 nM T09909 CBK6P1 11251114 Ki = 85 nM T09909 C1MVZ9 11251687 Ki > 10000 nM T09909 C5TQA4 11274375 Ki = 32 nM T09909 CA9X7I 11296725 Ki = 17 nM T09909 CJ7ZW8 11297638 Ki > 10000 nM T09909 CY8I0M 11316477 Ki = 70 nM T09909 CJL09Y 11317806 Ki = 0.5 nM T09909 CCU1Y4 11331355 Ki > 10000 nM T09909 CC8E0W 11331641 Ki = 48 nM T09909 C8KIU9 11341901 Ki > 10000 nM T09909 C6C4ND 11365721 Ki = 133 nM T09909 CH5F3D 11366289 Ki = 46 nM T09909 CU7A9K 11373911 Ki > 10000 nM T09909 CN8TX4 11378160 Ki > 10000 nM T09909 CB3EV8 11407509 Ki > 10000 nM T09909 CX3AQ4 11411528 Ki > 10000 nM T09909 C9SYG3 11422958 Ki > 10000 nM T09909 C4Q1ZA 11445913 Ki = 37.4 nM T09909 CQ5I1T 11467611 Ki > 10000 nM T09909 CV2E4Z 11476710 IC50 = 10000 nM T09909 CEC50O 11490141 Ki > 10000 nM T09909 CIT91Y 11564291 Ki = 1.85 nM T09909 C9G6ND 11672486 Ki = 9.8 nM T09909 C16ORL 11722069 Ki = 41.3 nM T09909 CSQ3P5 11758341 IC50 = 549 nM T09909 CDGF69 11765177 IC50 = 2 nM T09909 CD7E5Q 11765454 IC50 = 20 nM T09909 C9I0HX 11765560 IC50 = 2.5 nM T09909 C6QYM2 11766283 Ki = 10.1 nM T09909 CL1Q9G 11994156 Ki = 6 nM T09909 C7O8WN 11994288 Ki > 10000 nM T09909 CJ47YL 11994289 Ki = 0.6 nM T09909 C2MG6C 11994290 Ki = 2 nM T09909 CHQ72N 11994291 Ki = 0.5 nM T09909 C32DBH 11994292 Ki = 15 nM T09909 CP2GJ1 11994293 Ki = 34 nM T09909 CJ19TK 11995654 Ki > 10000 nM T09909 CER83M 11995655 Ki = 4 nM T09909 CW39RU 11995658 Ki = 189 nM T09909 CFGH32 13996286 Ki = 0.9 nM T09909 C40VIG 15171724 IC50 = 0.13 nM T09909 CQZ71Y 15222070 IC50 = 700 nM T09909 CG5XH2 15222092 IC50 = 80 nM T09909 CBPL06 15222094 IC50 = 600 nM T09909 CO5V6R 15222101 IC50 = 600 nM T09909 CO71QD 15222103 IC50 = 500 nM T09909 CZV27T 15230312 IC50 = 59 nM T09909 COW6H2 15230313 IC50 = 9.4 nM T09909 CL95MD 15230315 IC50 = 370 nM T09909 CY6TC4 15230316 IC50 = 730 nM T09909 CE7L9K 15284887 IC50 = 5.1 nM T09909 CF57HL 15292111 IC50 = 9.2 nM T09909 CX75ZV 15292112 IC50 = 9.8 nM T09909 CG29NO 15292113 IC50 = 3.3 nM T09909 CYS18L 15296723 IC50 = 70 nM T09909 C1PS5Y 15296724 IC50 = 1100 nM T09909 C5BDP4 15296725 IC50 = 150 nM T09909 C83KVY 15296726 IC50 = 750 nM T09909 CT09GK 15698118 IC50 = 140 nM T09909 CSK27N 15818746 IC50 = 300 nM T09909 CV40ST 15818748 IC50 = 100 nM T09909 C3TG8P 16087340 Ki = 53.1 nM T09909 CZ5CF4 16087341 Ki = 4.7 nM T09909 CARE54 16087342 Ki = 1.8 nM T09909 CMP48E 16124926 Ki > 10000 nM T09909 CL42BE 16124927 Ki > 10000 nM T09909 CT9XC2 16124928 Ki = 40.6 nM T09909 C27DCQ 16124929 Ki = 37.5 nM T09909 CU24SQ 16725318 IC50 = 260 nM T09909 CAG89Z 19102815 IC50 = 270 nM T09909 C8BLT0 19430442 IC50 = 1.6 nM T09909 CVL4G0 19430458 IC50 = 2.1 nM T09909 C60YHR 19430462 IC50 = 1.9 nM T09909 CRC30I 19430475 IC50 = 0.69 nM T09909 CVF5K9 19430479 IC50 = 0.9 nM T09909 CL86JK 19742811 IC50 = 2 nM T09909 CRC8L6 19763341 IC50 = 6.7 nM T09909 CZO2D5 19802473 IC50 = 2.3 nM T09909 C2KQ7M 19939495 IC50 = 140 nM T09909 C4O6AC 20647138 IC50 = 0.89 nM T09909 C8JR6C 22402420 IC50 = 4.8 nM T09909 CAU8T1 22402428 IC50 = 170 nM T09909 C84JSP 22402431 IC50 = 35 nM T09909 CMX5K3 22402433 IC50 = 40 nM T09909 CB1JC2 22402434 IC50 = 1.9 nM T09909 CG2D3I 23583071 IC50 = 102 nM T09909 C80VNF 23584461 IC50 = 1120 nM T09909 C1A5RE 23666226 IC50 = 920 nM T09909 CQPD98 23683656 IC50 = 0.58 nM T09909 CIG6B0 25135102 IC50 = 78 nM T09909 CE69MC 44210864 IC50 = 200 nM T09909 CL8Y6H 44212339 Ki = 4.5 nM T09909 CY4MC9 44283372 IC50 = 30 nM T09909 C07SPU 44299561 IC50 = 80 nM T09909 CB20ZQ 44299632 IC50 = 12 nM T09909 CG3L2O 44299633 IC50 = 7.4 nM T09909 CD85YE 44299634 IC50 = 0.82 nM T09909 CS6FW1 44299646 IC50 = 6.1 nM T09909 C2A7PO 44299647 IC50 = 4.8 nM T09909 CZSU59 44299655 IC50 = 0.47 nM T09909 C9LEX4 44299671 IC50 = 9.1 nM T09909 C8YBR1 44299731 IC50 = 1.74 nM T09909 CJ4V0Q 44299747 IC50 = 28 nM T09909 C2MS7P 44299748 IC50 = 27 nM T09909 C5A0KR 44299820 IC50 = 0.65 nM T09909 C5P1LM 44299845 IC50 = 86 nM T09909 C4MH6O 44311071 IC50 = 10 nM T09909 C04OWQ 44311072 IC50 = 1 nM T09909 CVXU13 44311073 IC50 = 3 nM T09909 C64VDR 44311074 IC50 = 7 nM T09909 C3O6SW 44311182 IC50 = 3 nM T09909 CCD7K5 44311183 IC50 = 3 nM T09909 CDC7V8 44311184 IC50 = 3 nM T09909 CYSE79 44311185 IC50 = 3 nM T09909 CFO20B 44311289 IC50 = 2 nM T09909 C5FI1X 44311342 IC50 = 600 nM T09909 CHW83V 44311406 IC50 = 200 nM T09909 C37PFG 44311412 IC50 = 1 nM T09909 CAK8C2 44311413 IC50 = 2 nM T09909 CHJP87 44311414 IC50 = 2 nM T09909 C3WZY9 44311415 IC50 = 5 nM T09909 COTX54 44311428 IC50 = 300 nM T09909 C8C5HR 44311429 IC50 = 600 nM T09909 CW7V8A 44311434 IC50 = 2 nM T09909 CT6A4H 44311435 IC50 = 2 nM T09909 C7FH8G 44311436 IC50 = 9 nM T09909 C5P6NM 44311449 IC50 > 10000 nM T09909 CWVO75 44311450 IC50 = 1000 nM T09909 CL68EO 44311451 IC50 = 70 nM T09909 C3H1MD 44311452 IC50 = 1 nM T09909 C3F6SU 44311453 IC50 = 20 nM T09909 C6Q0UC 44311454 IC50 = 9 nM T09909 C7SD4Z 44311455 IC50 = 2 nM T09909 CKT0U8 44311456 IC50 = 4 nM T09909 C5HPL4 44311472 IC50 = 7000 nM T09909 C23KJT 44311496 IC50 = 100 nM T09909 C9CY1G 44311497 IC50 = 1000 nM T09909 CC9Y6E 44311498 IC50 = 80 nM T09909 CL9Z1B 44311499 IC50 = 200 nM T09909 CRF13T 44311537 IC50 = 3 nM T09909 CKI10X 44311538 IC50 = 10 nM T09909 COI20G 44311543 IC50 = 400 nM T09909 C4FAK2 44311557 IC50 = 20 nM T09909 CB41MY 44311558 IC50 = 20 nM T09909 C3X1AL 44311567 IC50 = 1000 nM T09909 CY7DG6 44311568 IC50 = 800 nM T09909 C1XC8Q 44311569 IC50 = 400 nM T09909 CD4ZM5 44311571 IC50 = 1000 nM T09909 C5UBK7 44311580 IC50 = 3 nM T09909 CX90KA 44311581 IC50 = 5 nM T09909 CT05AS 44311582 IC50 = 5 nM T09909 CUAI35 44311583 IC50 = 300 nM T09909 CTP18U 44311584 IC50 = 200 nM T09909 C04GME 44311607 IC50 = 4000 nM T09909 C0R6QJ 44311609 IC50 = 300 nM T09909 C5LJ8A 44311616 IC50 = 2000 nM T09909 CSH0R1 44311617 IC50 = 10 nM T09909 C92KSW 44311618 IC50 = 5 nM T09909 CPGV60 44311619 IC50 = 3 nM T09909 CSE80D 44311635 IC50 = 200 nM T09909 C6CQ3Y 44311636 IC50 = 500 nM T09909 CLT7J0 44311638 IC50 = 500 nM T09909 CXZ1Y2 44311648 IC50 = 700 nM T09909 CX89YT 44311650 IC50 = 90 nM T09909 CU4HB9 44311662 IC50 = 90 nM T09909 C0I8FS 44311663 IC50 = 400 nM T09909 CT1X8Z 44311664 IC50 = 1000 nM T09909 CR7Q4V 44311675 IC50 = 1 nM T09909 C3X7ZI 44311676 IC50 = 1 nM T09909 C8SY2D 44311681 IC50 = 3000 nM T09909 C46NML 44311683 IC50 = 5 nM T09909 CP7CY2 44311688 IC50 = 6000 nM T09909 CJ9A7D 44311715 IC50 = 2 nM T09909 C07CUQ 44311735 IC50 = 3 nM T09909 CBW43X 44311736 IC50 = 1 nM T09909 CPX02A 44311738 IC50 > 10000 nM T09909 CJ2N1I 44311739 IC50 = 90 nM T09909 CA1Y6I 44311752 IC50 = 10 nM T09909 CAB87G 44311753 IC50 = 2 nM T09909 C8VU6N 44311754 IC50 = 2 nM T09909 C8UXN7 44311755 IC50 = 10 nM T09909 CFZE67 44311758 IC50 = 300 nM T09909 C29QVB 44311775 IC50 = 3000 nM T09909 CKF7H2 44311776 IC50 = 2000 nM T09909 CLV28B 44314761 IC50 = 4.4 nM T09909 CUIL91 44314780 IC50 = 6.5 nM T09909 CD28FL 44314822 IC50 = 7.8 nM T09909 CJS04N 44314823 IC50 = 7.7 nM T09909 CXDG91 44315057 IC50 = 12.5 nM T09909 C6XVW9 44315058 IC50 = 11 nM T09909 C08CHF 44315059 IC50 = 37 nM T09909 C4VD7T 44315060 IC50 = 32 nM T09909 C2JM6E 44315078 IC50 = 8 nM T09909 CF89XK 44315144 IC50 = 3.5 nM T09909 C8S9UP 44315180 IC50 = 12 nM T09909 CH0ZF3 44315282 IC50 = 8.9 nM T09909 C1STV6 44315304 IC50 = 9.3 nM T09909 CTD3M0 44315344 IC50 = 11 nM T09909 CJ4SK0 44315349 IC50 = 65 nM T09909 C8QAE0 44315350 IC50 = 65 nM T09909 CH9Q0J 44315351 IC50 = 3.1 nM T09909 CI6OR9 44321626 IC50 = 3500 nM T09909 C1W4SY 44321775 IC50 = 8.2 nM T09909 CP75AN 44321790 IC50 = 5 nM T09909 CSDL17 44321791 IC50 = 1.1 nM T09909 CFT1B9 44321804 IC50 = 9.1 nM T09909 CL3UZ9 44321823 IC50 = 5.6 nM T09909 CJ7Y3T 44321824 IC50 = 1.9 nM T09909 CPC59Y 44321825 IC50 = 3.9 nM T09909 CNY2L4 44322095 IC50 = 2 nM T09909 C6JRB7 44322096 IC50 = 4.7 nM T09909 CM6TB8 44322097 IC50 = 15 nM T09909 CP34OW 44322176 IC50 = 8 nM T09909 CLJ1H4 44322202 IC50 = 1.1 nM T09909 C0Q5PE 44322203 IC50 = 1.1 nM T09909 CPHC67 44322233 IC50 = 44 nM T09909 C3G8PO 44322234 IC50 = 38 nM T09909 CN2C4V 44322235 IC50 = 3800 nM T09909 C3RI8C 44322236 IC50 = 120 nM T09909 C3W0UX 44348523 IC50 = 1.7 nM T09909 CBHM56 44365273 IC50 = 0.08 nM T09909 CJR05U 44371045 IC50 = 5.8 nM T09909 CSO26P 44372686 IC50 = 24 nM T09909 CTRJ86 44372814 IC50 = 180 nM T09909 CQ46VS 44373238 IC50 = 12 nM T09909 CVW3K2 44377942 IC50 = 100 nM T09909 CG0F2S 44381883 Ki = 0.62 nM T09909 C0RJ4U 44382994 IC50 = 7 nM T09909 COWV95 44398242 Ki = 1 nM T09909 C3GOI4 44398381 Ki = 3.7 nM T09909 C97XTV 44400615 Ki = 9.3 nM T09909 CU8D4I 44400670 Ki = 2.8 nM T09909 CI8HL6 44404967 IC50 = 32 nM T09909 CE5HS1 44417234 Ki = 0.7 nM T09909 C1XCM5 44420766 Ki > 10000 nM T09909 C51DFM 44420768 Ki = 1110 nM T09909 CGK9O3 44420769 Ki > 10000 nM T09909 C47HPS 44420771 Ki > 10000 nM T09909 C62TGK 44420773 Ki > 10000 nM T09909 C5WJO4 44420774 Ki > 10000 nM T09909 C2CYT9 44420775 Ki = 16.6 nM T09909 C3GYC0 44475943 IC50 = 5070 nM T09909 CCG7X8 44574325 IC50 = 850 nM T09909 C65RAJ 45102601 Ki = 2511.89 nM T09909 CG3B8F 45102750 Ki > 10000 nM T09909 CBAG18 46910582 IC50 = 1200 nM T09909 CF7ID9 46910583 IC50 = 1500 nM T09909 C6SAG5 56657702 Ki = 2.6 nM T09909 C71ABG 56661223 Ki = 0.08 nM T09909 CIDV38 56678310 Ki = 61 nM T09909 C9DMZ4 56964910 Ki = 17.8 nM T09909 C20CLX 57380412 IC50 = 1100 nM T09909 CG09ZX 57380413 IC50 > 10000 nM T09909 C19NLI 57380414 IC50 = 3600 nM T09909 CQ5IJ3 57380415 IC50 > 10000 nM T09909 C2AVN8 57380416 IC50 > 10000 nM T09909 CZRA28 57380647 IC50 = 1400 nM T09909 C52XFK 57380649 IC50 = 1300 nM T09909 C1L5WH 60148656 IC50 = 4366 nM T09909 CN9MK3 71455883 IC50 = 25 nM T09909 CF20NM 73213175 Ki = 42000 nM T09909 CV8JL5 73213176 Ki = 18000 nM T09909 CQ0WC6 73213177 Ki > 100000 nM T09909 CT9E3S 73213178 Ki = 29000 nM T09909 CC0AG8 73213179 Ki = 8500 nM T09909 CM1Z2I 73213180 Ki = 9200 nM T09909 C35QZR 73213252 Ki = 9900 nM T09909 CPT05L 73213253 Ki > 100000 nM T09909 CML1C7 73213255 Ki > 100000 nM T09909 C9YX2T 73213256 Ki > 100000 nM T09909 CS3I2T 73346386 IC50 > 10000 nM T09909 C5L6PQ 73347892 IC50 = 78 nM T09909 C4COR6 73347893 IC50 = 149 nM T09909 CEOK17 73349424 IC50 = 42 nM T09909 C2LTU4 73350991 IC50 > 10000 nM T09909 C9ZC5N 73353933 IC50 = 718 nM T09909 CG71DK 73353934 IC50 = 53 nM T09909 CRGQ95 73355474 IC50 > 10000 nM T09909 CCEA97 73355475 IC50 = 77 nM T09909 CB9DV4 73357016 IC50 = 6 nM T09909 CU53JN 73357017 IC50 = 164 nM T09909 C6HJS2 73357018 IC50 = 61 nM T09909 CW0J4R 76313892 Ki = 47000 nM T09909 CZ2I6V 76324571 IC50 > 10000 nM T09909 C6UG1S 90663955 IC50 = 116 nM T09909 C80FBU 118719020 Ki = 0.7 nM T09909 CC9DI5 118725967 Ki = 12.3 nM T09909 CB1XJ0 118725969 Ki = 8.2 nM T09909 CKB0S3 136059719 IC50 = 190 nM T09909 CECL48 136059720 IC50 < 10 nM T09909 CIJ5E0 136059721 IC50 = 250 nM T09909 C5P3ZF 145963801 Ki = 130 nM T09909 CLH9Q6 145964638 Ki = 390 nM T09909 CMY82H 145965035 Ki = 730 nM T09909 CKY1Q9 145965121 Ki = 160 nM T09909 CB4S2Z 145965943 Ki = 480 nM T09909 CQ1ZK5 145966800 Ki = 440 nM T09909 C7O5YA 145967796 Ki = 270 nM T09909 CNS37J 145969149 Ki = 290 nM T09909 CBTD16 145972310 Ki = 2300 nM T09909 CDP0L2 145972801 Ki = 400 nM T09909 CB9U4F 145972980 Ki = 400 nM T09909 C79OXW 145974498 Ki = 300 nM T09909 C8SCF2 145976243 Ki = 280 nM T09909 CUH5J9 145976532 Ki = 340 nM T09909 C2CXD0 145977406 Ki = 180 nM T09909 CG8MY6 145978135 Ki = 140 nM T09909 CV3L9X 145978497 Ki = 230 nM T09909 CIRC08 145978684 Ki = 300 nM T09909 CC9V8J 44382947 IC50 = 3.6 nM T09909 D04SVT 9829012 IC50 = 4500 nM T09909 D09FRL 114899 IC50 = 66 nM T09909 D0A4NO 6603900 IC50 = 2 nM T09909 D0K2EX 9804984 Ki = 0.4 nM T09909 D0M5ZE 5311416 Ki < 10000 nM T09909 D0OF3M 10373777 Ki = 0.18 nM T09909 D0Z7AF 10031067 IC50 = 0.7 nM T66252 D02EYG 10096344 IC50 = 100000 nM T66252 D0K9MY 11243969 Ki = 71 nM T66252 D0L3DK 6918537 Ki = 68 nM T66252 D0NJ5H 11450633 IC50 > 100000 nM T66252 D0T8XB 44513473 IC50 = 60 nM T66252 D0U2JP 4369359 IC50 = 3060 nM T66252 D04XIO 11253490 IC50 = 663 nM T66252 D07EPV 11949652 IC50 = 540 nM T66252 D07HZG 11516136 IC50 = 5980 nM T66252 D0FQ2U 6918572 Ki = 0.76 nM T66252 D0M3XR 46209133 IC50 > 67000 nM T66252 D04MAZ 71731606 IC50 > 100000 nM T66252 D0A1NU 16049769 Ki > 30000 nM T66252 D0F3TI 11673176 Ki = 2.6 nM T66252 D0Q4YP 11996845 IC50 = 60000 nM T66252 CE98OF 6451150 IC50 = 20000 nM T66252 CCIX30 9209502 IC50 = 168 nM T66252 C14VRG 9794073 IC50 = 2100 nM T66252 CSA6V9 9796352 IC50 = 13700 nM T66252 C62DNH 9843297 IC50 > 100000 nM T66252 CZUQ34 9883487 IC50 = 320 nM T66252 C2TV9M 9884543 IC50 = 86 nM T66252 C28XTC 9942425 IC50 > 100000 nM T66252 CQ8J7T 9953181 IC50 > 100000 nM T66252 CT6XQ2 9983092 IC50 = 25000 nM T66252 C78NMY 10026124 IC50 > 100000 nM T66252 C83ZDL 10096130 IC50 = 1400 nM T66252 C0Q7BK 10127057 IC50 > 100000 nM T66252 C2H0UF 10149048 Ki = 0.53 nM T66252 C4CX1P 10157141 IC50 > 100000 nM T66252 C5P0AO 10238227 IC50 > 100000 nM T66252 CZ90LD 10250452 IC50 = 69000 nM T66252 CU8C5K 10254918 IC50 > 100000 nM T66252 C17HUN 10255762 IC50 > 100000 nM T66252 C6ER9U 10269517 IC50 = 3200 nM T66252 C3FB4T 10310021 IC50 = 53000 nM T66252 CF1S8U 10320144 IC50 > 100000 nM T66252 CNV4R3 10324641 IC50 > 100000 nM T66252 CM6Y1B 10339570 Ki = 23000 nM T66252 C7UO3L 10376704 Ki > 30000 nM T66252 CQ7J2Z 10383508 IC50 > 100000 nM T66252 CY5M4R 10388027 IC50 = 43000 nM T66252 C29MEL 10399628 Ki > 30000 nM T66252 CVK1G5 10412922 IC50 = 28000 nM T66252 C80ZBS 10429788 IC50 > 100000 nM T66252 C6GHF1 10433039 IC50 > 100000 nM T66252 CWCA76 10439426 IC50 > 86000 nM T66252 CAF71Y 10443207 IC50 = 28000 nM T66252 C4OC6P 10455620 IC50 = 20000 nM T66252 C1WKE4 10455621 IC50 = 62000 nM T66252 CH1DG5 10478099 IC50 = 54000 nM T66252 CK3IW4 10584272 IC50 = 11200 nM T66252 C0KTQ5 10607253 IC50 > 100000 nM T66252 CHA8X6 10751333 IC50 = 50000 nM T66252 CYLO09 10774283 IC50 > 50000 nM T66252 CL26WQ 10780092 IC50 > 100000 nM T66252 C2KDY6 10798619 IC50 > 100000 nM T66252 C1WG0P 10798659 IC50 = 2 nM T66252 C1ZJ4I 10799226 IC50 = 16000 nM T66252 CJKX61 10821833 IC50 = 76000 nM T66252 C7BLJ1 10821834 IC50 > 100000 nM T66252 C3E8ID 10845163 IC50 = 38400 nM T66252 CK9SB4 10845727 IC50 > 100000 nM T66252 CLA05J 10932707 Ki = 3300 nM T66252 CA4N0B 11117606 Ki = 293 nM T66252 CF1LD8 11199808 Ki = 505 nM T66252 C68XFD 11205761 IC50 > 1000000 nM T66252 CHX25W 11232123 IC50 > 100000 nM T66252 CYL67P 11232890 Ki = 107 nM T66252 CKL1A8 11268930 Ki = 49 nM T66252 CM0YI7 11269397 Ki = 73 nM T66252 C5IY0L 11269712 IC50 > 100000 nM T66252 C2SOA8 11306467 IC50 > 100000 nM T66252 C47GSV 11310499 IC50 = 5100 nM T66252 CEZ27P 11314348 Ki = 39 nM T66252 CTG12Q 11321743 IC50 > 100000 nM T66252 CNB7G8 11356095 IC50 = 5100 nM T66252 CKP0G9 11362130 IC50 = 80 nM T66252 CW3QZ7 11374531 IC50 > 100000 nM T66252 C30JEU 11381416 IC50 > 30000 nM T66252 CL9HN3 11395030 Ki = 60 nM T66252 CTW02K 11406276 Ki = 300 nM T66252 CRZ5F1 11418876 IC50 > 100000 nM T66252 CY15PU 11429829 Ki = 50 nM T66252 CH09SE 11447824 IC50 = 26400 nM T66252 CWO06L 11471453 IC50 = 2500 nM T66252 C7JWD3 11476287 IC50 > 100000 nM T66252 CS4H7X 11481506 IC50 = 118 nM T66252 CTD0S4 11486251 Ki = 1777 nM T66252 CNMA97 11487118 IC50 > 100000 nM T66252 C06RUA 11493219 IC50 > 30000 nM T66252 CDT16S 11493492 Ki > 30000 nM T66252 CJD30Y 11495704 IC50 = 3700 nM T66252 CAH5Z6 11500899 IC50 > 30000 nM T66252 CH7VS5 11505454 IC50 = 1700 nM T66252 CM8QB3 11510166 Ki > 10000 nM T66252 C2S8BH 11516511 Ki > 30000 nM T66252 CH5A7Q 11518007 IC50 = 2600 nM T66252 C2TCM8 11523077 IC50 = 5500 nM T66252 C8KB4F 11524437 Ki > 30000 nM T66252 CMYN65 11526865 IC50 > 100000 nM T66252 C0O3XD 11527019 IC50 > 100000 nM T66252 CZFI65 11531704 Ki = 3100 nM T66252 C1B8JN 11532057 Ki > 30000 nM T66252 CZ35WN 11533932 IC50 > 100000 nM T66252 COXK41 11537890 Ki > 30000 nM T66252 CK36XC 11538961 Ki = 9800 nM T66252 CG7I8Z 11538992 IC50 > 100000 nM T66252 CPR71X 11540951 IC50 > 100000 nM T66252 C98GDW 11541277 IC50 > 100000 nM T66252 CBR9K8 11541314 IC50 > 100000 nM T66252 C6KBN4 11546261 Ki = 2.2 nM T66252 C2DJ6Y 11552953 Ki > 30000 nM T66252 CA16WP 11554165 IC50 = 38000 nM T66252 CDK7I5 11559922 Ki = 3.3 nM T66252 CI5W4Y 11566450 IC50 > 30000 nM T66252 CR37GC 11567606 Ki = 1 nM T66252 CY0A7J 11570138 IC50 > 100000 nM T66252 CAE39I 11573427 IC50 > 30000 nM T66252 CE03TL 11574811 Ki > 10000 nM T66252 CQU80H 11576569 IC50 > 100000 nM T66252 CW94NS 11577331 IC50 > 100000 nM T66252 CQ86GI 11577431 IC50 > 100000 nM T66252 CAZL49 11584650 IC50 > 100000 nM T66252 C5JYV7 11591936 IC50 > 100000 nM T66252 CO0QJ8 11596007 Ki > 30000 nM T66252 CE8M3K 11596123 Ki > 30000 nM T66252 C9MXO0 11596219 IC50 > 20000 nM T66252 CBE6K8 11603637 Ki = 5600 nM T66252 CPXV24 11603996 IC50 > 100000 nM T66252 C15DLO 11608317 IC50 = 800 nM T66252 COF62W 11611325 Ki > 10000 nM T66252 CQL5S8 11613750 IC50 > 100000 nM T66252 CD3YU1 11616861 IC50 > 30000 nM T66252 C2APG7 11623550 IC50 > 30000 nM T66252 CRY2D5 11625412 Ki = 5800 nM T66252 C7YKC0 11628195 IC50 > 100000 nM T66252 CSO1D6 11632159 Ki > 30000 nM T66252 CM1DR9 11632375 Ki > 20000 nM T66252 CHLA97 11638762 Ki > 30000 nM T66252 CRA0H5 11639131 Ki > 30000 nM T66252 CQO8U6 11648011 Ki > 30000 nM T66252 CXG1B4 11649741 IC50 > 100000 nM T66252 CZBD50 11653749 Ki > 30000 nM T66252 C94OMG 11654093 Ki > 30000 nM T66252 C8AU5P 11654528 Ki = 5500 nM T66252 C52ION 11655271 Ki > 30000 nM T66252 CCBS09 11674180 Ki > 30000 nM T66252 CTNO72 11674721 IC50 = 11000 nM T66252 C2G6RP 11675637 Ki = 7800 nM T66252 CI1ED9 11676224 IC50 = 15000 nM T66252 C3Y7EL 11678025 IC50 = 14000 nM T66252 C7DCV9 11696495 Ki > 30000 nM T66252 C6JPE0 11696912 Ki > 30000 nM T66252 CRU2Q1 11697286 Ki = 2100 nM T66252 C2WK1Z 11697387 Ki = 4500 nM T66252 C2X5GC 11704411 Ki = 4800 nM T66252 C6YHK3 11704412 Ki = 5900 nM T66252 CK4I6J 11710700 Ki > 30000 nM T66252 C04OMI 11711314 Ki > 30000 nM T66252 C8VC2D 11711413 Ki > 30000 nM T66252 C8KD6N 11711414 Ki = 5300 nM T66252 C34BEP 11716483 Ki > 30000 nM T66252 C1XD5I 11718004 Ki > 30000 nM T66252 CIEJ54 11720809 IC50 > 100000 nM T66252 C6JY7V 11776638 Ki > 30000 nM T66252 C6ET2R 11817181 IC50 = 76900 nM T66252 CQIB43 11957945 IC50 > 100000 nM T66252 C6BHJ9 15101668 IC50 > 100000 nM T66252 C2ZMH8 15948988 IC50 = 3735 nM T66252 C13JIX 15949418 IC50 = 45400 nM T66252 C49NUJ 15949507 IC50 = 72300 nM T66252 CU4P5X 15950383 Ki = 1097 nM T66252 C16XRI 15950384 Ki > 30000 nM T66252 CUMR27 15950385 Ki = 971 nM T66252 C69RAY 15950386 Ki = 2313 nM T66252 CM63YP 15950387 Ki = 5860 nM T66252 CH8F7W 15950388 Ki = 1057 nM T66252 C0L4SH 15950456 Ki > 30000 nM T66252 C8G7OJ 15950457 Ki = 2298 nM T66252 C9KJ6D 15950538 Ki = 3439 nM T66252 C3C6PM 15950539 Ki = 2938 nM T66252 C4S7AB 15950540 Ki = 2830 nM T66252 C2HGJ0 15950541 Ki = 2637 nM T66252 C3U1VO 15950542 Ki > 30000 nM T66252 CKX8M6 15950615 Ki > 30000 nM T66252 CC0M2X 15951427 Ki = 3840 nM T66252 CF3PX0 15951428 Ki = 8511 nM T66252 CWTX01 15951429 Ki = 1461 nM T66252 C3LQD9 15951431 Ki = 2233 nM T66252 CI3DB4 15951636 IC50 = 2700 nM T66252 CL1E6O 15953860 IC50 > 100000 nM T66252 CLG2Q1 16035093 IC50 = 32000 nM T66252 CMUG74 16035094 IC50 = 58000 nM T66252 C13-MAR 16040457 IC50 > 100000 nM T66252 CS7DQ3 16090844 Ki > 30000 nM T66252 C8CVG9 16090856 Ki > 30000 nM T66252 CU3GB5 16126742 IC50 = 710.7 nM T66252 CHUX72 16202788 Ki > 3000 nM T66252 CC20IT 16203037 Ki > 3000 nM T66252 CA1PV5 16216352 IC50 > 20000 nM T66252 C53XZP 16721117 Ki > 3000 nM T66252 CT01PQ 16739331 IC50 = 48977.88 nM T66252 C61RFP 16755651 IC50 = 9420 nM T66252 CU05RG 17748274 IC50 > 100000 nM T66252 C5W3VY 17753031 IC50 > 100000 nM T66252 CT42AI 20706081 IC50 = 13900 nM T66252 C0X4SO 22029457 IC50 > 100000 nM T66252 CLK4G6 22029894 IC50 > 100000 nM T66252 CED47V 22690988 IC50 = 68100 nM T66252 C8JSI4 23628284 IC50 = 100000 nM T66252 CAQ81M 23644660 IC50 > 100000 nM T66252 CDPU25 23644665 IC50 > 100000 nM T66252 CCSU21 23645371 IC50 = 330 nM T66252 CFV07G 23645410 IC50 > 100000 nM T66252 CIMG82 23645411 IC50 > 100000 nM T66252 C2Q5IK 23645581 IC50 = 2720 nM T66252 C3VA0M 23645582 IC50 > 100000 nM T66252 C4B9FM 23645685 Ki = 3 nM T66252 CP9GS5 23645686 IC50 > 100000 nM T66252 C6R2LP 23645687 IC50 > 100000 nM T66252 CN7FK3 23645688 IC50 > 100000 nM T66252 CSHX17 23645689 IC50 > 100000 nM T66252 CL8QV6 23645690 IC50 > 100000 nM T66252 C0AU9X 23645691 IC50 > 100000 nM T66252 CRM3Y4 23645692 IC50 > 100000 nM T66252 CDM8A2 23645693 IC50 > 100000 nM T66252 CIR1F6 23645694 IC50 > 100000 nM T66252 CK5G6I 23645695 IC50 > 100000 nM T66252 CHS76O 23645696 IC50 > 100000 nM T66252 CVP59D 23645697 IC50 > 100000 nM T66252 CH13BW 23645698 IC50 > 100000 nM T66252 CL0K1T 23645699 IC50 > 100000 nM T66252 CB3Z7O 23645700 IC50 > 100000 nM T66252 CNO6Q1 23645702 IC50 > 100000 nM T66252 CGMC54 23645703 IC50 > 100000 nM T66252 C0V4WR 23645705 IC50 > 100000 nM T66252 CKM6Y8 23645917 IC50 = 63000 nM T66252 C9Y2ZL 23645918 IC50 = 65000 nM T66252 C4V6BX 23645919 IC50 > 100000 nM T66252 C78PNU 23645920 IC50 > 100000 nM T66252 C5YT6S 23645921 IC50 > 100000 nM T66252 CELQ89 23645922 IC50 > 100000 nM T66252 CGV92H 23645923 IC50 = 24000 nM T66252 CJ60EH 23645924 IC50 = 27000 nM T66252 CZG70A 23645925 IC50 > 100000 nM T66252 CD6V7X 23645926 IC50 > 100000 nM T66252 C1TD4J 23645927 IC50 > 100000 nM T66252 C71PQU 23645928 IC50 = 50000 nM T66252 C8EOB9 23645929 IC50 > 100000 nM T66252 C0M1TH 23645930 IC50 > 100000 nM T66252 CFHB36 23645931 IC50 > 100000 nM T66252 CTG27F 23645932 IC50 = 13000 nM T66252 CS2FT5 23645933 IC50 = 26000 nM T66252 C98QGK 23645934 IC50 = 34000 nM T66252 CS76DY 23645935 IC50 > 100000 nM T66252 C91MYK 23645936 IC50 = 36000 nM T66252 C3AQC0 23645937 IC50 > 100000 nM T66252 C61GTC 23645938 IC50 = 20000 nM T66252 C8XF6R 23645939 IC50 = 41000 nM T66252 C7IX5B 23645940 IC50 = 7800 nM T66252 CP6M3W 23645941 IC50 = 9600 nM T66252 CQ75XK 23645942 IC50 = 5100 nM T66252 C8T7GY 23645943 IC50 = 6500 nM T66252 C25ZXC 23645944 IC50 = 30000 nM T66252 C4A3NI 23645945 IC50 > 100000 nM T66252 CVSH12 23646026 IC50 = 53 nM T66252 CZ28UC 23646142 Ki > 30000 nM T66252 CLA15H 23646143 Ki = 10 nM T66252 CDM3J0 23646514 Ki > 3000 nM T66252 CBA8N1 23647136 IC50 = 98000 nM T66252 CVF6E2 23661697 IC50 > 100000 nM T66252 CM7C4W 23661708 IC50 = 43000 nM T66252 CO6L9F 23661716 IC50 = 19000 nM T66252 CHR14F 23661718 IC50 > 100000 nM T66252 CNP9T1 24180585 IC50 > 30000 nM T66252 C0H8OB 24776705 IC50 > 100000 nM T66252 C24GLZ 24776939 IC50 = 20000 nM T66252 C6LD2J 24777439 IC50 > 100000 nM T66252 CK8EL5 24777568 IC50 = 52000 nM T66252 CQ20PV 24777692 IC50 > 100000 nM T66252 C1WF3I 24777804 IC50 > 100000 nM T66252 C29SZR 24784416 IC50 = 240 nM T66252 CY9W8O 24860300 IC50 = 13000 nM T66252 CMK9B7 24894026 IC50 = 70 nM T66252 CX83WL 24963343 IC50 > 100000 nM T66252 CA94RD 24999327 IC50 = 5700 nM T66252 CZJ2N6 24999330 IC50 = 5040 nM T66252 C01GPL 25132159 Ki = 2100 nM T66252 C7IDX9 25132160 Ki = 50 nM T66252 C9VK8W 25132161 Ki = 260 nM T66252 CFZ4V2 25132162 Ki = 4300 nM T66252 CSU0B5 25189891 Ki > 30000 nM T66252 C7KN2U 42608447 IC50 = 5100 nM T66252 CS40ML 44123747 IC50 > 50000 nM T66252 CQF86D 44182505 IC50 = 2430 nM T66252 C3I4TF 44201003 IC50 > 50000 nM T66252 CE5B7H 44218404 IC50 > 20000 nM T66252 CR8GT4 44218550 IC50 > 20000 nM T66252 CBW7D4 44218551 IC50 > 20000 nM T66252 CISE95 44218553 IC50 > 20000 nM T66252 CLB72R 44218554 IC50 > 20000 nM T66252 C2N9VR 44218555 IC50 > 20000 nM T66252 CJ6L3S 44218693 IC50 > 20000 nM T66252 C97IFE 44218695 IC50 > 20000 nM T66252 C50EKW 44250174 IC50 = 2900 nM T66252 CFY7P3 44360924 IC50 = 570 nM T66252 CPX1M9 44403336 IC50 = 65 nM T66252 CSEN70 44403337 IC50 = 510 nM T66252 C0NXE8 44403338 IC50 = 43000 nM T66252 C91MNA 44403353 IC50 = 800 nM T66252 CR53EK 44403354 IC50 = 400 nM T66252 C8MLN6 44403355 IC50 = 280 nM T66252 CRO16Q 44403360 IC50 = 4.6 nM T66252 C0FC7D 44403361 IC50 = 6.7 nM T66252 CCOA39 44403438 IC50 = 220 nM T66252 CLYJ80 44403439 IC50 = 160 nM T66252 CSG4F8 44417393 Ki = 1760 nM T66252 C59HZQ 44418251 IC50 = 6500 nM T66252 C0FT8Q 44420999 Ki > 30000 nM T66252 C6NV0S 44421004 Ki = 18300 nM T66252 C5W8VX 44421005 Ki = 19700 nM T66252 C9IRG5 44422418 IC50 = 501.1 nM T66252 CS63GZ 44422443 IC50 = 518.9 nM T66252 CNQC83 44422485 IC50 = 748.7 nM T66252 C7IL3S 44431164 IC50 > 100000 nM T66252 C0UOS8 44431165 IC50 > 100000 nM T66252 CEG05S 44431166 IC50 > 100000 nM T66252 CO8S3Z 44431170 IC50 > 100000 nM T66252 C2K4RQ 44431176 IC50 > 100000 nM T66252 CJZY21 44431177 IC50 > 100000 nM T66252 CSJI40 44431185 IC50 > 100000 nM T66252 C36EJR 44431188 IC50 > 100000 nM T66252 C2MCA1 44431191 IC50 > 100000 nM T66252 C89XVB 44431197 IC50 > 100000 nM T66252 CK76EP 44431199 IC50 > 100000 nM T66252 C3FPT2 44431200 IC50 > 100000 nM T66252 C4F8AG 44431201 IC50 = 72000 nM T66252 CWX4I3 44431203 IC50 > 100000 nM T66252 CZ3N9E 44431204 IC50 = 49000 nM T66252 C5NAS6 44431205 IC50 > 100000 nM T66252 C37SGU 44431206 IC50 > 100000 nM T66252 CYD62G 44431212 IC50 > 100000 nM T66252 C72WTP 44431213 IC50 > 58000 nM T66252 CC3T9G 44431214 IC50 > 100000 nM T66252 CL4T3X 44431215 IC50 > 78000 nM T66252 C4WVL8 44431216 IC50 > 100000 nM T66252 CO08HZ 44431217 IC50 > 100000 nM T66252 CCPZ23 44431218 IC50 > 100000 nM T66252 C0J7WV 44431219 IC50 > 100000 nM T66252 C16ZTV 44431220 IC50 = 78000 nM T66252 CR0A1M 44431316 IC50 > 100000 nM T66252 CV1R7A 44431317 IC50 > 100000 nM T66252 C9GIE3 44433617 IC50 > 100000 nM T66252 C5B4HS 44433618 IC50 = 3100 nM T66252 CU6XZ5 44433646 IC50 = 40000 nM T66252 CM8E2D 44433661 IC50 = 50000 nM T66252 CEL4H9 44439337 IC50 = 30 nM T66252 C0OJ1T 44439353 IC50 = 110 nM T66252 C08ZST 44440659 Ki > 3000 nM T66252 CR3PM7 44440662 Ki = 17500 nM T66252 CB4Q0H 44440663 Ki = 10900 nM T66252 CCSI57 44440665 Ki = 11100 nM T66252 CA0NZ7 44443707 IC50 = 51000 nM T66252 C24ZHB 44443708 IC50 > 100000 nM T66252 C8R4OD 44443709 IC50 = 50000 nM T66252 CLDN63 44443710 IC50 > 100000 nM T66252 C7LNP2 44443711 IC50 = 63000 nM T66252 CJX2M7 44443712 IC50 > 100000 nM T66252 C6RST0 44443713 IC50 > 100000 nM T66252 C3YL9X 44443714 IC50 > 100000 nM T66252 CRH8M1 44443715 IC50 > 100000 nM T66252 CIB50E 44443717 IC50 = 9400 nM T66252 CK6QF4 44443719 IC50 = 73000 nM T66252 CX6O1P 44443720 IC50 > 100000 nM T66252 C0YV2D 44443723 IC50 = 89000 nM T66252 C1BUJ5 44443725 IC50 = 15000 nM T66252 CXS34I 44443727 IC50 > 100000 nM T66252 CCHS17 44443729 IC50 > 100000 nM T66252 CS3Y1G 44444344 IC50 > 100000 nM T66252 CL2U9C 44444352 IC50 > 100000 nM T66252 C8VE5T 44444353 IC50 > 100000 nM T66252 C8F5HC 44444371 IC50 = 27000 nM T66252 CEW50M 44444373 IC50 = 27000 nM T66252 CO0M7Y 44444375 IC50 = 54000 nM T66252 CS93BI 44444377 IC50 > 100000 nM T66252 C9J4FB 44444379 IC50 > 100000 nM T66252 C3YA4K 44444383 IC50 = 77000 nM T66252 C75OIP 44444386 IC50 = 27000 nM T66252 C4J6ZG 44444390 IC50 > 100000 nM T66252 C05EBU 44444391 IC50 > 100000 nM T66252 CSN27E 44445042 IC50 = 26000 nM T66252 CGN61Q 44445047 IC50 = 41000 nM T66252 CYW8E3 44445051 IC50 > 100000 nM T66252 CRG64M 44445053 IC50 = 24000 nM T66252 C6ZID3 44445055 IC50 = 18000 nM T66252 C72KOR 44445057 IC50 > 100000 nM T66252 C0RTA6 44445060 IC50 = 39000 nM T66252 CIK8G3 44445063 IC50 = 89000 nM T66252 CN05VX 44445065 IC50 > 100000 nM T66252 COA90R 44445067 IC50 > 100000 nM T66252 C91DWY 44560396 IC50 = 8600 nM T66252 CZ9WJ0 44560397 IC50 > 100000 nM T66252 C0FLU7 44560398 IC50 = 540 nM T66252 CX9BK6 44560399 IC50 = 88 nM T66252 CZ43JR 44560454 IC50 = 7600 nM T66252 CY38QP 44560549 IC50 > 100000 nM T66252 C7IL3K 44560550 IC50 > 100000 nM T66252 CF9J7Z 44560551 IC50 = 4100 nM T66252 C1QAI4 44560552 IC50 > 50000 nM T66252 CK25CG 44560553 IC50 > 25000 nM T66252 C4C9NG 44560554 IC50 = 96000 nM T66252 CKIH45 44560555 IC50 = 82800 nM T66252 C2LW3C 44560595 IC50 = 1200 nM T66252 C47WCK 44560596 IC50 = 1100 nM T66252 CL8AE5 44560597 IC50 > 100000 nM T66252 C1YJ8C 44560648 IC50 = 200 nM T66252 CY6GU1 44560649 IC50 = 2390 nM T66252 C12EYZ 44560650 IC50 = 169 nM T66252 C7LY9V 44560651 IC50 = 3670 nM T66252 CG5CB2 44560698 IC50 = 13100 nM T66252 CR56BA 44560699 IC50 = 41000 nM T66252 CIA45R 44560700 IC50 = 16100 nM T66252 CAK3U5 44560701 IC50 = 5770 nM T66252 CJE42H 44560746 IC50 = 6690 nM T66252 C5OW2C 44560747 IC50 = 67800 nM T66252 CM2GN5 44560748 IC50 = 29800 nM T66252 C5FSB4 44560749 IC50 > 25000 nM T66252 C5WEG1 44560750 IC50 = 2650 nM T66252 CZSO82 44560823 IC50 = 34200 nM T66252 C4IVD9 44560824 IC50 = 62400 nM T66252 C4L3VZ 44560825 IC50 = 2790 nM T66252 CHV7S1 44560826 IC50 = 14500 nM T66252 CE3NF4 44560849 IC50 = 10900 nM T66252 CTH9P2 44560851 IC50 = 15900 nM T66252 C9EK8A 44560929 IC50 > 100000 nM T66252 CM68VD 44560930 IC50 = 1420 nM T66252 C4SMJ1 44560961 IC50 = 212 nM T66252 C2I3TR 44560962 IC50 = 35 nM T66252 CGV49L 44560963 IC50 = 6.3 nM T66252 CY0L1G 44560964 IC50 = 25 nM T66252 CGOM86 44560989 IC50 = 9200 nM T66252 C74ZNK 44560990 IC50 = 82 nM T66252 C95AUS 44560991 IC50 = 4.6 nM T66252 CRO3D2 44567651 IC50 = 547 nM T66252 CM95OD 44567652 IC50 = 5990 nM T66252 CD4C7Y 44567710 IC50 = 63200 nM T66252 C4CUJ6 44567711 IC50 = 350 nM T66252 CK1C7W 44567712 IC50 = 525 nM T66252 CTK1I9 44567713 IC50 = 7300 nM T66252 CM50CU 44567747 IC50 = 2410 nM T66252 CNA0I9 44567918 IC50 = 421 nM T66252 C6BXT0 44567919 IC50 = 131 nM T66252 CJ85MG 44567920 IC50 = 1660 nM T66252 CUJD19 44567976 IC50 = 343 nM T66252 C5YB6E 44567977 IC50 = 66 nM T66252 CNF09E 44567978 IC50 = 807 nM T66252 C70WEI 44567979 IC50 = 130 nM T66252 CW7NB6 44568016 IC50 = 771 nM T66252 CY8Z3F 44568017 IC50 = 640 nM T66252 CRM76D 44568018 IC50 = 3030 nM T66252 CCG83U 44568057 IC50 = 729 nM T66252 C8XW9A 44568058 IC50 = 119 nM T66252 CMQ7D5 44568097 IC50 = 1910 nM T66252 C1F9OL 44568098 IC50 = 169 nM T66252 CUYK75 44568099 IC50 = 1910 nM T66252 CZ81XF 44568100 IC50 = 3680 nM T66252 C6GT0A 44568134 IC50 = 4850 nM T66252 C6IW5D 44568135 IC50 = 1960 nM T66252 C3PWD8 44568136 IC50 = 1200 nM T66252 C4NCA7 44568169 IC50 > 100000 nM T66252 C8TXH9 44568170 IC50 = 5420 nM T66252 C17PZX 44568171 IC50 = 448 nM T66252 C7SCJ1 44568172 IC50 = 7810 nM T66252 C2DQ0C 44589933 IC50 = 9000 nM T66252 CUZ3P0 44589935 IC50 = 37600 nM T66252 CBAH06 44590649 IC50 = 100 nM T66252 CRN4U5 44590696 IC50 > 100000 nM T66252 CY8R3Q 44593399 IC50 = 4300 nM T66252 CP8YC3 44593408 IC50 = 500 nM T66252 C65KPR 45101722 IC50 = 3700 nM T66252 CXYT36 45101723 IC50 = 3900 nM T66252 C2RNP7 45102670 IC50 = 27000 nM T66252 CGZD98 45265711 IC50 > 100000 nM T66252 CW09DZ 45265891 Ki > 3000 nM T66252 CCO76A 45266134 IC50 > 100000 nM T66252 CU4C5P 45266135 IC50 = 100000 nM T66252 CLVM20 45266136 IC50 > 100000 nM T66252 C8H9GV 45267527 IC50 = 1400 nM T66252 CP9B0W 45267530 IC50 = 350 nM T66252 C3GJK0 45267531 IC50 = 2700 nM T66252 CN38QU 45268229 IC50 = 3400 nM T66252 CEQ16V 45268233 IC50 = 100 nM T66252 C0QB1V 45268417 IC50 = 1700 nM T66252 C2S9ZT 45268436 IC50 = 1300 nM T66252 CX8WC0 45269123 IC50 = 2500 nM T66252 C9HR0K 45269274 IC50 = 2700 nM T66252 CZ1N2O 45269275 IC50 = 1100 nM T66252 CIE21V 45269276 IC50 = 470 nM T66252 CWT60M 45269971 IC50 = 8800 nM T66252 C8QJ7X 45270108 IC50 = 1700 nM T66252 CYWK62 45270115 IC50 = 4000 nM T66252 CGF7Z6 45270958 IC50 = 1700 nM T66252 CH5S8Y 45270959 IC50 = 5000 nM T66252 C5NH6Q 45271791 IC50 = 990 nM T66252 C8Z3DK 45271794 IC50 = 3000 nM T66252 CX62YA 45271796 IC50 = 4400 nM T66252 CZ8EO2 45271803 IC50 = 3600 nM T66252 CJ7Q9E 45271813 IC50 = 1200 nM T66252 CJI2R6 45272664 IC50 = 1100 nM T66252 C49BKQ 45272672 IC50 = 2000 nM T66252 CP36CT 45272682 IC50 = 880 nM T66252 C8NL4U 45272683 IC50 = 1600 nM T66252 C6S0OC 45273404 IC50 = 1200 nM T66252 CYMR87 45273573 IC50 = 1200 nM T66252 CFL87A 45273581 IC50 = 1200 nM T66252 C2XB0P 45273589 IC50 = 1500 nM T66252 C28PRV 45273594 IC50 = 3200 nM T66252 CSX2T9 45273602 IC50 = 15000 nM T66252 CMP59Q 45273603 IC50 = 1500 nM T66252 C28ZXW 45487888 IC50 = 24000 nM T66252 C2N3IZ 45487894 IC50 = 11000 nM T66252 CP62TC 45487898 IC50 = 5100 nM T66252 CWQ1R9 45487903 IC50 = 7400 nM T66252 C8H1KY 45487904 IC50 = 4800 nM T66252 C6X7WJ 45487908 IC50 = 6600 nM T66252 C5OXM9 45487915 IC50 = 12000 nM T66252 CPJ19X 45487917 IC50 = 27000 nM T66252 CV2R7M 45487920 IC50 = 8200 nM T66252 C57JRG 45487921 IC50 = 17000 nM T66252 C4JD1P 45487922 IC50 = 36000 nM T66252 CPB85R 45487926 IC50 = 19000 nM T66252 CTY16E 45487930 IC50 = 17000 nM T66252 C4QTL9 45487931 IC50 = 9800 nM T66252 CG9V0L 45487940 IC50 = 14000 nM T66252 C5XTV1 45487945 IC50 = 910 nM T66252 C3VK4G 45487946 IC50 = 1600 nM T66252 CDP7Q4 46870369 IC50 = 2740 nM T66252 CPH7B4 46871723 IC50 = 37 nM T66252 CDBC45 46890720 IC50 > 20000 nM T66252 CLK47C 46890721 IC50 > 20000 nM T66252 CS6HL3 46890722 IC50 > 20000 nM T66252 C2JY6P 46890723 IC50 > 20000 nM T66252 CP7C1L 46890780 IC50 > 20000 nM T66252 CA3PE4 46890853 IC50 > 20000 nM T66252 CY9T8W 46890854 IC50 > 20000 nM T66252 CT9HQ6 46890913 IC50 > 20000 nM T66252 CSZE87 46891193 IC50 = 3220 nM T66252 C18UES 46891235 IC50 = 1400 nM T66252 C23LCY 46891237 IC50 = 6860 nM T66252 C57UXS 46891239 IC50 = 7750 nM T66252 CJ4G6X 46891342 IC50 = 1380 nM T66252 CPN5T2 46891535 IC50 > 20000 nM T66252 C4XTW7 46893990 IC50 > 50000 nM T66252 C8O5VR 46899592 Ki > 30 nM T66252 CTY0M5 46899593 Ki = 1.9 nM T66252 CK9TH1 46899594 Ki = 1.3 nM T66252 C8XD0Q 46899595 Ki = 2.2 nM T66252 CZ84ST 46899596 Ki = 0.83 nM T66252 CPZ70E 46899597 Ki = 2 nM T66252 CD3IJ8 46899752 Ki = 0.9 nM T66252 CRK59N 46899753 Ki = 3.5 nM T66252 C6LXU5 46899754 Ki = 2.5 nM T66252 C52JZL 46899755 Ki = 0.94 nM T66252 C4RC1S 46899756 Ki = 5.8 nM T66252 CP84HR 46899757 Ki = 2.5 nM T66252 CBV4W0 46899937 Ki = 0.6 nM T66252 C5QEJ4 46899938 Ki = 0.9 nM T66252 CHR6V9 46899939 Ki = 3.5 nM T66252 CQ3A8F 46899940 Ki = 5.6 nM T66252 CX2P8Z 46899941 Ki = 0.55 nM T66252 CC2X1J 46899942 Ki = 0.86 nM T66252 C5QA9M 46900103 Ki = 3.5 nM T66252 C4IU2E 46900105 Ki = 1.9 nM T66252 CZEB71 46900106 Ki = 3.3 nM T66252 C2TJW5 46900108 Ki = 0.3 nM T66252 C54ATK 46900259 Ki = 2.1 nM T66252 CI3P6J 46900261 Ki = 1.4 nM T66252 C6DP2G 46900418 Ki = 1.5 nM T66252 CP50DR 46900420 Ki > 10 nM T66252 C8DSG7 46916343 IC50 > 100000 nM T66252 C3RO8F 46916345 IC50 > 100000 nM T66252 CX07LJ 46916346 IC50 > 100000 nM T66252 CF94MW 46916347 IC50 > 100000 nM T66252 CH3F7O 46916384 IC50 > 20000 nM T66252 CM8W6E 46916385 IC50 > 100000 nM T66252 C6FA9Q 46916386 IC50 > 20000 nM T66252 CAW86J 46916387 IC50 > 100000 nM T66252 C63HBE 46916388 IC50 > 100000 nM T66252 CD1CZ7 46916389 IC50 > 100000 nM T66252 CH80LK 46916433 IC50 > 50000 nM T66252 CN4A3P 46916435 IC50 > 100000 nM T66252 CUQ86M 46917047 IC50 > 50000 nM T66252 CS5X9L 46917048 IC50 > 100000 nM T66252 CZP24U 46917049 IC50 = 520 nM T66252 CGMJ52 46938499 IC50 > 100000 nM T66252 C5RAS7 46938602 IC50 > 100000 nM T66252 C3B1LX 46938704 IC50 > 50000 nM T66252 C5TU1F 46938705 IC50 > 100000 nM T66252 CAGP83 46938706 IC50 > 20000 nM T66252 CP9V8Q 46938799 IC50 > 100000 nM T66252 CAB2H9 46938802 IC50 > 100000 nM T66252 C80RAT 47370344 IC50 > 100000 nM T66252 CR5X3K 49785099 IC50 > 25000 nM T66252 C2HU0V 49785100 IC50 > 25000 nM T66252 CX7M2K 49785101 IC50 > 25000 nM T66252 C3XCV4 49785102 IC50 > 25000 nM T66252 CZ7A9E 49796933 IC50 > 100000 nM T66252 C5RF0Y 49796938 IC50 = 450 nM T66252 CE0C3Y 49796939 IC50 > 100000 nM T66252 CI4ZE6 49796940 IC50 = 71000 nM T66252 CBD8K2 49796942 IC50 > 100000 nM T66252 CI25XP 49796945 IC50 > 100000 nM T66252 C8WYA5 49796953 IC50 = 86000 nM T66252 CQH86V 49796955 IC50 > 100000 nM T66252 CBMV50 49796972 IC50 = 86000 nM T66252 C8IL0K 49796973 IC50 > 100000 nM T66252 CA90LB 49796974 IC50 > 100000 nM T66252 C07DHG 49796977 IC50 > 100000 nM T66252 CAS2P4 49796982 IC50 > 100000 nM T66252 CG79KT 49796985 IC50 > 100000 nM T66252 C4D8RE 49796990 IC50 > 100000 nM T66252 CUKB68 49796994 IC50 > 100000 nM T66252 CUR9B0 49796995 IC50 = 62000 nM T66252 CWHO58 49796998 IC50 > 100000 nM T66252 CX74RG 49796999 IC50 = 69000 nM T66252 C20MAQ 49797000 IC50 > 100000 nM T66252 CD67OX 49797001 IC50 > 100000 nM T66252 C9LEF5 49797002 IC50 = 26000 nM T66252 CO2AX9 49797003 IC50 = 2600 nM T66252 CEM61W 49797006 IC50 > 100000 nM T66252 C7Y0JL 49797007 IC50 > 100000 nM T66252 CW45IK 49797008 IC50 > 100000 nM T66252 C79JUI 49797011 IC50 > 100000 nM T66252 CVAK94 49797012 IC50 > 100000 nM T66252 CUK5J1 49797013 IC50 = 57000 nM T66252 C4ZK5C 49797014 IC50 > 100000 nM T66252 C1PV8J 49797015 IC50 > 100000 nM T66252 C9YEU6 49797016 IC50 > 100000 nM T66252 CZD4S2 49797017 IC50 > 100000 nM T66252 CKY80F 49797018 IC50 > 100000 nM T66252 CS0D8Q 49797021 IC50 = 46000 nM T66252 C3GF4M 49797022 IC50 > 100000 nM T66252 C8XZT9 49797023 IC50 > 100000 nM T66252 C5H2AS 49797024 IC50 > 100000 nM T66252 C4P0VW 49797025 IC50 > 100000 nM T66252 CVY8M1 49797028 IC50 > 100000 nM T66252 CM59HB 49797029 IC50 > 100000 nM T66252 CH7Y1J 49797030 IC50 > 100000 nM T66252 CX18HI 49797031 IC50 = 81000 nM T66252 CUM28Z 49797035 IC50 > 100000 nM T66252 COS23G 49797036 IC50 = 66000 nM T66252 C2TSG6 49797038 IC50 > 100000 nM T66252 C7BI3W 49797039 IC50 > 100000 nM T66252 C71THK 49797040 IC50 > 100000 nM T66252 C0SG5O 49797041 IC50 > 100000 nM T66252 CM37VB 49797042 IC50 > 100000 nM T66252 C51NUG 49797043 IC50 > 100000 nM T66252 C65WXC 49797044 IC50 > 100000 nM T66252 CHTO37 49797045 IC50 > 100000 nM T66252 CA8R5K 49797046 IC50 > 100000 nM T66252 CLAR35 49797047 IC50 > 100000 nM T66252 C9OCZ3 49797048 IC50 > 100000 nM T66252 C49RUW 49797049 IC50 = 78000 nM T66252 C4EHT7 49797050 IC50 > 100000 nM T66252 CW6G5R 49797051 IC50 = 34000 nM T66252 CUK6G0 49797052 IC50 > 100000 nM T66252 CJ1FE2 49797053 IC50 = 95000 nM T66252 CKJO08 49797054 IC50 > 100000 nM T66252 C70KVU 49797055 IC50 > 100000 nM T66252 CP59BI 49797056 IC50 = 67000 nM T66252 CEDL61 49797057 IC50 > 100000 nM T66252 C5J2LV 49797058 IC50 > 100000 nM T66252 CEI20Q 49797059 IC50 > 100000 nM T66252 C7B5DY 49797060 IC50 = 52000 nM T66252 C5B1RM 49797061 IC50 > 100000 nM T66252 C40HJC 49797062 IC50 > 100000 nM T66252 CL3P4H 49797063 IC50 > 100000 nM T66252 CPC76U 49797064 IC50 > 100000 nM T66252 C5F4JN 49797065 IC50 > 100000 nM T66252 C86HND 49797066 IC50 > 100000 nM T66252 C8E4XD 49797067 IC50 > 100000 nM T66252 CHO1U0 49797068 IC50 = 37000 nM T66252 CO1TW7 49797069 IC50 > 100000 nM T66252 CAD6W1 49797071 IC50 = 57000 nM T66252 CQYU80 49797072 IC50 > 100000 nM T66252 CEZ38H 49797073 IC50 > 100000 nM T66252 C0CEU7 49797074 IC50 > 100000 nM T66252 C72JXY 49797075 IC50 = 59000 nM T66252 COA41Q 49797076 IC50 > 100000 nM T66252 CPQ3Z2 49797077 IC50 > 100000 nM T66252 C1WI0D 49797078 IC50 = 48000 nM T66252 C4D8XP 49797079 IC50 > 100000 nM T66252 CQG4J6 49797080 IC50 > 100000 nM T66252 CKM9S4 49797081 IC50 > 100000 nM T66252 C3JRW0 49797082 IC50 > 100000 nM T66252 C27IEB 49797083 IC50 > 100000 nM T66252 C0JUL3 49797084 IC50 = 45000 nM T66252 C85DOL 49797085 IC50 > 100000 nM T66252 CEGO30 49797086 IC50 > 100000 nM T66252 C2TC3I 49797087 IC50 > 100000 nM T66252 C04JWY 49797088 IC50 = 79000 nM T66252 CA2U4Y 49797089 IC50 > 100000 nM T66252 CFT46J 49797090 IC50 > 100000 nM T66252 C35TFW 49797091 IC50 > 100000 nM T66252 CRL7Z5 49797092 IC50 > 100000 nM T66252 CYU74X 49797093 IC50 > 100000 nM T66252 C2O3SG 49797094 IC50 > 100000 nM T66252 CFL3O2 49797106 IC50 > 100000 nM T66252 CF4NR7 49797107 IC50 > 100000 nM T66252 CV9QW6 49797108 IC50 > 100000 nM T66252 CJZA65 49797109 IC50 > 100000 nM T66252 CBS36X 49797110 IC50 > 100000 nM T66252 C0STP5 49797111 IC50 > 100000 nM T66252 C7KV5R 49797112 IC50 > 100000 nM T66252 CJPX53 49797113 IC50 > 100000 nM T66252 C2OI0Y 49797114 IC50 > 100000 nM T66252 CW20FJ 49797115 IC50 > 100000 nM T66252 C9P6VU 49797116 IC50 > 100000 nM T66252 C67SIA 49797117 IC50 > 100000 nM T66252 CCI8Y0 49797118 IC50 > 100000 nM T66252 CE10UF 49797119 IC50 > 100000 nM T66252 CLH0V3 49797120 IC50 = 59000 nM T66252 C2N8WX 49797121 IC50 > 100000 nM T66252 CNCE06 49797122 IC50 > 100000 nM T66252 C76UAB 49797123 IC50 > 100000 nM T66252 CHWT89 49797124 IC50 > 100000 nM T66252 C1Z6NE 49797125 IC50 > 100000 nM T66252 C25MQG 49797126 IC50 > 100000 nM T66252 COL54B 49797127 IC50 > 100000 nM T66252 C5OUQ3 49797128 IC50 > 100000 nM T66252 C3NMI8 49797173 Ki = 73 nM T66252 C1E3YB 49797174 Ki = 500 nM T66252 CVD0I1 49797175 Ki = 430 nM T66252 CH02OC 49797176 Ki = 14000 nM T66252 CY1OJ5 49797177 Ki = 4000 nM T66252 C25ZSD 49797191 IC50 > 100000 nM T66252 C0OJX9 49797192 IC50 > 100000 nM T66252 C7GZ4B 49797193 IC50 > 100000 nM T66252 CVT2E5 49797194 IC50 > 100000 nM T66252 C75MGE 49797195 IC50 > 100000 nM T66252 CVS70C 49797196 IC50 > 100000 nM T66252 C42QPW 49797197 IC50 > 100000 nM T66252 C6ZGL5 49797198 IC50 > 100000 nM T66252 C1B5NH 49797199 IC50 > 100000 nM T66252 CGQN24 49797200 IC50 > 100000 nM T66252 CS2AI5 49797201 IC50 > 100000 nM T66252 CM7RE3 49797202 IC50 > 100000 nM T66252 CGM9E7 49797203 IC50 > 100000 nM T66252 COU0I6 49797204 IC50 > 100000 nM T66252 C3XML2 49797205 IC50 > 100000 nM T66252 CP0O2F 49797223 IC50 = 39000 nM T66252 CTH7I8 49797224 IC50 = 38000 nM T66252 CG9P7O 49797225 IC50 = 36000 nM T66252 C3A2QK 49797226 IC50 = 35000 nM T66252 C4NOK2 49797227 IC50 = 21000 nM T66252 CB13PO 49797228 IC50 = 13000 nM T66252 C47VOG 49797229 IC50 > 100000 nM T66252 CD2CL1 49797230 IC50 > 100000 nM T66252 C0LK6B 49797231 IC50 = 9600 nM T66252 CON0A6 49797232 IC50 = 67000 nM T66252 C4AVU3 49797233 IC50 = 58000 nM T66252 CQ93MI 49797234 IC50 = 40000 nM T66252 CO2JV8 49797235 IC50 = 44000 nM T66252 C27LDC 49797236 IC50 = 13000 nM T66252 CA5GM6 49797237 IC50 > 100000 nM T66252 CT8PW1 49797238 IC50 = 50000 nM T66252 CJQ38S 49797239 IC50 = 37000 nM T66252 CT65MR 49797240 IC50 > 100000 nM T66252 C08IFZ 49797241 IC50 > 100000 nM T66252 CA4E8M 49797242 IC50 > 100000 nM T66252 CN8FR2 49797243 IC50 = 75000 nM T66252 C37MDP 49797244 IC50 > 100000 nM T66252 CM41RN 49797245 IC50 = 57000 nM T66252 C59JEK 49797246 IC50 = 32000 nM T66252 CUMH43 49797248 IC50 > 100000 nM T66252 CM59PE 49797249 IC50 > 100000 nM T66252 CN5K1S 49797250 IC50 > 100000 nM T66252 CT5HY0 49797251 IC50 = 91000 nM T66252 C0E5PY 49797252 IC50 = 90000 nM T66252 C3E5JB 49797253 IC50 > 100000 nM T66252 CA8P5N 49797344 IC50 > 100000 nM T66252 CJL2B8 49797345 IC50 > 100000 nM T66252 CT79YI 49797346 IC50 > 100000 nM T66252 C93VJO 49797347 IC50 > 100000 nM T66252 CDI52A 49797348 IC50 > 100000 nM T66252 C7ATK9 49797349 IC50 > 100000 nM T66252 C2Y3DS 49797350 IC50 > 100000 nM T66252 CA4CE3 49797351 IC50 > 100000 nM T66252 C3A8YT 49797352 IC50 > 100000 nM T66252 C1Z8HB 49797353 IC50 = 2700 nM T66252 CC0T8H 49797354 IC50 > 100000 nM T66252 C92QND 49797355 IC50 = 42000 nM T66252 C2HPE8 49797356 IC50 > 100000 nM T66252 C9UXH2 49797357 IC50 = 26000 nM T66252 CTYO37 49797358 IC50 > 100000 nM T66252 C1K4FR 49797359 IC50 = 46000 nM T66252 CJ2D0P 49797360 IC50 = 63000 nM T66252 CA3Q2W 49797361 IC50 > 100000 nM T66252 CNMF62 49797362 IC50 = 29000 nM T66252 CU72EZ 49797596 IC50 = 79000 nM T66252 C6AZ2C 49797599 IC50 > 100000 nM T66252 CR86PO 49797604 IC50 = 60000 nM T66252 C6DJX7 49797605 IC50 > 100000 nM T66252 CK3ZI1 49797607 IC50 = 63000 nM T66252 C7AD0C 49797610 IC50 > 100000 nM T66252 C4XHO5 49797612 IC50 > 100000 nM T66252 C7VL5U 49797614 IC50 = 73000 nM T66252 CY09JE 49797615 IC50 = 81000 nM T66252 C1ZLF0 49797616 IC50 > 100000 nM T66252 CN48OE 49797627 IC50 = 71000 nM T66252 CV6I0O 49797630 IC50 > 100000 nM T66252 CAG1U7 49797631 IC50 > 100000 nM T66252 C8JNU1 49797636 IC50 > 100000 nM T66252 C0DN5G 49797642 IC50 = 60000 nM T66252 CJVS96 49797644 IC50 > 100000 nM T66252 CBRT78 49797650 IC50 > 100000 nM T66252 CZW93Y 49797653 IC50 > 100000 nM T66252 COM5Q7 49836030 IC50 > 10000 nM T66252 CTDR85 49862539 Ki > 30000 nM T66252 CT8Q9N 49862713 Ki > 30000 nM T66252 C0OB8C 49862714 Ki > 30000 nM T66252 CJ58AG 49862715 Ki > 30000 nM T66252 C42TSR 49862716 Ki > 30000 nM T66252 CPU7F6 49862790 Ki > 30000 nM T66252 C4FZY2 49862791 Ki > 30000 nM T66252 CF40YM 49862792 Ki > 30000 nM T66252 CK0GC5 49864113 Ki = 0.28 nM T66252 CK1CD3 50925423 IC50 > 10000 nM T66252 C7T6PI 50994092 IC50 = 30000 nM T66252 C67CTP 51032641 IC50 > 25000 nM T66252 CL4S9Y 51050450 IC50 > 30000 nM T66252 CLU39H 51051131 IC50 = 30000 nM T66252 C5PRF8 51051132 IC50 = 12000 nM T66252 CYF04M 51051134 IC50 = 2400 nM T66252 CPCY75 51051136 IC50 = 1600 nM T66252 C7JM3I 51051236 IC50 = 11000 nM T66252 CZ5HJ0 51051238 IC50 = 3000 nM T66252 C1OUG5 51051240 IC50 = 5800 nM T66252 C6GAP9 51051329 IC50 > 30000 nM T66252 C9KPJ6 51051331 IC50 > 100000 nM T66252 C85CEJ 51346970 IC50 > 100000 nM T66252 C4PFT3 51346971 IC50 = 16000 nM T66252 C4VC2U 52942435 IC50 > 10000 nM T66252 C2B6EX 52943488 Ki > 10000 nM T66252 C56CXU 52943631 IC50 > 10000 nM T66252 CHD7O6 52943758 IC50 > 10000 nM T66252 C4I6ML 52944843 IC50 > 10000 nM T66252 C57XSM 52944845 IC50 > 10000 nM T66252 CT6SQ3 52944941 IC50 > 10000 nM T66252 C7RJM9 52945660 IC50 = 89 nM T66252 C9OAF1 52946149 IC50 > 10000 nM T66252 CC56BV 52946866 IC50 > 50000 nM T66252 CC7N8S 52948914 IC50 > 10000 nM T66252 C4LVO6 52948971 IC50 > 10000 nM T66252 CTU0J1 52949742 IC50 > 10000 nM T66252 CEFX05 53311069 IC50 > 100000 nM T66252 CQL50R 53311070 IC50 > 100000 nM T66252 C1Q4WK 53311071 IC50 > 100000 nM T66252 C67LHZ 53311072 IC50 > 100000 nM T66252 CQ0ZJ2 53311073 IC50 > 100000 nM T66252 C7PMY1 53311074 IC50 > 100000 nM T66252 CWN9H7 53311140 IC50 > 100000 nM T66252 CAL51C 53311141 IC50 > 100000 nM T66252 C2SXV0 53311142 IC50 > 100000 nM T66252 C7AEF8 53311143 IC50 > 100000 nM T66252 C5IOZ6 53311144 IC50 > 100000 nM T66252 CVR4H3 53311222 IC50 > 100000 nM T66252 CNX08H 53311223 IC50 > 100000 nM T66252 CET6W5 53311225 IC50 > 100000 nM T66252 C3RZS4 53311226 IC50 > 100000 nM T66252 CHR17Y 53311227 IC50 > 100000 nM T66252 C3HGW8 53312238 IC50 > 100000 nM T66252 CM03UX 53312239 IC50 > 100000 nM T66252 C9K4CZ 53312243 IC50 > 100000 nM T66252 CU4BS2 53312323 IC50 > 100000 nM T66252 CF5I6O 53312326 IC50 > 100000 nM T66252 C6PSL2 53312327 IC50 > 100000 nM T66252 C0WYS5 53312328 IC50 > 100000 nM T66252 CYC69Q 53317564 IC50 = 47000 nM T66252 C0QOV9 53317565 IC50 = 30000 nM T66252 CURC70 53317566 IC50 > 100000 nM T66252 C3ZK1W 53317575 IC50 = 12000 nM T66252 CBQ0J7 53317579 IC50 = 14000 nM T66252 CIY9F7 53317580 IC50 = 16000 nM T66252 C5DMS9 53317581 IC50 > 100000 nM T66252 C1XD9W 53317582 IC50 = 25000 nM T66252 CR0O8T 53317583 IC50 = 27000 nM T66252 C9GLH7 53318841 IC50 = 28000 nM T66252 C06TDE 53318842 IC50 = 32000 nM T66252 C73TER 53318856 IC50 = 57000 nM T66252 CC56NE 53318863 IC50 = 86000 nM T66252 C4UJI8 53318864 IC50 = 36000 nM T66252 C8CZ2A 53318865 IC50 = 7200 nM T66252 CLVY47 53318866 IC50 = 23000 nM T66252 CM7S5W 53319067 IC50 = 16000 nM T66252 C1X3NE 53320178 IC50 = 12000 nM T66252 C1P8BK 53320179 IC50 = 32000 nM T66252 C50UBZ 53320180 IC50 = 30000 nM T66252 C2JTR7 53320181 IC50 > 100000 nM T66252 C0TYJ5 53320182 IC50 = 18000 nM T66252 C7RSX2 53320183 IC50 = 12000 nM T66252 C9XGE4 53321472 IC50 = 61000 nM T66252 CY0ZV9 53321485 IC50 > 100000 nM T66252 CK0OB2 53321486 IC50 = 64000 nM T66252 CNK34J 53321487 IC50 = 85000 nM T66252 C7EO3D 53321495 IC50 = 13000 nM T66252 C3M7PQ 53321496 IC50 = 8100 nM T66252 C0NUQ7 53321497 IC50 = 12000 nM T66252 C31DSJ 53321498 IC50 = 19000 nM T66252 C2ZKV9 53321499 IC50 = 3100 nM T66252 C3QT0R 53321621 IC50 = 62000 nM T66252 CXIS21 53322758 IC50 = 76000 nM T66252 CY71QL 53322814 IC50 = 53000 nM T66252 CLU96Y 53322820 IC50 = 37000 nM T66252 C8YVF1 53322821 IC50 = 10000 nM T66252 C4QS6V 53322822 IC50 = 15000 nM T66252 C62JTB 53322823 IC50 = 17000 nM T66252 CT14FU 53322824 IC50 = 43000 nM T66252 CXJ1F8 53322825 IC50 = 24000 nM T66252 C3K1VY 53322826 IC50 = 19000 nM T66252 C9N6HK 53322952 IC50 = 77000 nM T66252 C9LU8M 53324129 IC50 = 31000 nM T66252 CCY7M0 53324130 IC50 = 24000 nM T66252 C4F1QK 53324142 IC50 > 100000 nM T66252 CZN71C 53324143 IC50 = 51000 nM T66252 CG83JZ 53324144 IC50 > 100000 nM T66252 CE8J1D 53324145 IC50 = 51000 nM T66252 C0Y3AC 53324153 IC50 = 81000 nM T66252 C9O1IW 53324154 IC50 = 45000 nM T66252 CTW5G0 53324155 IC50 = 59000 nM T66252 C2DPZ0 53324156 IC50 = 28000 nM T66252 CSN28M 53324293 IC50 > 100000 nM T66252 C25OJW 53325399 IC50 = 4200 nM T66252 CXW5O9 53325446 IC50 > 100000 nM T66252 C1SO0C 53325447 IC50 > 100000 nM T66252 C1S3WB 53325453 IC50 = 27000 nM T66252 C2KFW6 53325454 IC50 = 16000 nM T66252 C4ZFR5 53325455 IC50 = 23000 nM T66252 CV0H8P 53326691 IC50 = 27000 nM T66252 C3ZWN6 53326704 IC50 = 39000 nM T66252 C73SKG 53326705 IC50 = 55000 nM T66252 CG9V4W 53326706 IC50 = 16000 nM T66252 C5K8CP 53326713 IC50 > 100000 nM T66252 CN12AO 53353383 IC50 = 44000 nM T66252 C51GUC 53354365 IC50 > 100000 nM T66252 CRJ5P9 53354369 IC50 > 100000 nM T66252 C4G2HT 53354470 IC50 > 100000 nM T66252 CUC1N3 53356519 Ki = 5771 nM T66252 CSD1Q4 53357353 IC50 > 60000 nM T66252 C5UW0D 56652661 IC50 > 100000 nM T66252 C1QX0O 56657809 IC50 > 100000 nM T66252 C9OL5C 56962798 IC50 > 100000 nM T66252 CQX8J0 57385070 IC50 > 25000 nM T66252 CPS89B 57385071 IC50 > 25000 nM T66252 CNU9C0 57385072 IC50 > 10000 nM T66252 CG5MT6 57385073 IC50 > 10000 nM T66252 CQZ09L 57390626 IC50 = 53 nM T66252 CWR4E5 57390923 Ki = 1536 nM T66252 C0RAD8 57390924 Ki = 1890 nM T66252 C5U6RF 57392407 IC50 = 64 nM T66252 CD0OT2 57392409 IC50 = 66 nM T66252 C4QYJ6 57392724 Ki = 3496 nM T66252 CWDY79 57394441 Ki = 10490 nM T66252 CZ23RJ 57395915 IC50 = 81 nM T66252 C8KMS2 57396206 Ki = 262 nM T66252 C2QL6K 57397702 IC50 = 45 nM T66252 CBQ85O 57397704 IC50 = 30 nM T66252 C2ZE3R 57397706 IC50 = 21 nM T66252 CW97SN 57398006 Ki > 10000 nM T66252 C01KCU 57399665 Ki = 2430 nM T66252 C65ZFW 57401128 IC50 = 28 nM T66252 CYX43T 57401419 Ki = 5982 nM T66252 C1T0AD 57403169 Ki = 2340 nM T66252 C12QCM 57403170 Ki = 1101 nM T66252 CX94UQ 57403171 Ki = 1710 nM T66252 C1L8YD 57404359 IC50 = 3280 nM T66252 C8SX7A 57404360 IC50 = 2200 nM T66252 C0Q1OZ 57404374 IC50 > 50000 nM T66252 CL0UA1 57525787 IC50 = 105 nM T66252 C9ZE7J 58874273 IC50 > 100000 nM T66252 CZ4VD5 60032916 IC50 = 3.5 nM T66252 C9SND1 68305755 IC50 > 100000 nM T66252 CP3E2X 68416066 IC50 = 330 nM T66252 CCS6K9 68417211 IC50 = 610 nM T66252 C0C8JW 70293564 IC50 = 17600 nM T66252 CK26FY 70295607 IC50 > 30000 nM T66252 CV4X5S 70295927 IC50 = 13000 nM T66252 CXSV41 70296244 IC50 = 24600 nM T66252 C3SB1V 70296823 IC50 > 30000 nM T66252 CXD5V6 70297609 IC50 = 3500 nM T66252 CEG1L5 70330884 IC50 = 125 nM T66252 C5W6LY 70681316 IC50 = 53000 nM T66252 C97JFS 70682267 IC50 = 86 nM T66252 CE1FU2 70682268 IC50 = 40 nM T66252 C03SDB 70682493 IC50 = 2609 nM T66252 CF0U3A 70682494 IC50 = 4862 nM T66252 C8Z2UQ 70682495 IC50 = 2096 nM T66252 C4YW5T 70684349 IC50 = 180 nM T66252 C6W1CT 70684350 IC50 = 6900 nM T66252 C1GF3E 70684351 IC50 = 6.4 nM T66252 C1NHS4 70684571 IC50 = 4814 nM T66252 C1Q3ZO 70686506 IC50 = 2.1 nM T66252 C5I9BL 70686723 IC50 = 1368 nM T66252 CLQC52 70688610 IC50 = 35 nM T66252 CGQV87 70688811 IC50 = 471 nM T66252 CVYH31 70689717 IC50 = 23000 nM T66252 CYO5X6 70690674 IC50 = 14 nM T66252 C2J7FS 70690675 IC50 = 9.5 nM T66252 CL6KR9 70690676 IC50 = 0.31 nM T66252 CXE41O 70690893 IC50 = 658 nM T66252 C19FJC 70692822 IC50 = 200 nM T66252 C8JZ3Q 70692823 IC50 = 240 nM T66252 C3MF7C 70693037 IC50 = 2740 nM T66252 C5YQ9B 70693038 IC50 = 427 nM T66252 CEQ4N8 70693039 IC50 = 885 nM T66252 CYQO06 70693040 IC50 = 1449 nM T66252 CIX3F9 70694853 IC50 = 98 nM T66252 CQJD92 70694854 IC50 = 9.3 nM T66252 CA0W8R 70695074 IC50 = 318 nM T66252 CYB1P3 70695075 IC50 = 4746 nM T66252 C4ETL9 70695076 IC50 = 4226 nM T66252 C1NGL5 70696903 IC50 = 11 nM T66252 C2B5UF 70697122 IC50 = 1763 nM T66252 CJ4M0N 70697124 IC50 = 1013 nM T66252 C31UTS 71184301 IC50 = 14600 nM T66252 C8LY1U 71184352 IC50 > 30000 nM T66252 C9IRW7 71184590 IC50 > 30000 nM T66252 C08NDK 71184749 IC50 = 9000 nM T66252 CP91OE 71203742 IC50 > 100000 nM T66252 CP6G5W 71203746 IC50 > 100000 nM T66252 C32UMV 71203748 IC50 > 100000 nM T66252 C04XQY 71203752 IC50 > 100000 nM T66252 CE2I0K 71203758 IC50 > 100000 nM T66252 CIQ7O2 71203767 IC50 = 15828 nM T66252 C5GEJ9 71203769 IC50 > 100000 nM T66252 C7LKV0 71203783 IC50 > 100000 nM T66252 CP9K2W 71450603 IC50 = 1700 nM T66252 C61LNR 71452448 IC50 = 3000 nM T66252 CN4FE7 71454208 IC50 = 7000 nM T66252 C1LRH5 71455960 IC50 = 11200 nM T66252 C59TGZ 71457761 IC50 = 7700 nM T66252 C5T6QP 71457765 IC50 = 17400 nM T66252 CUB4V8 71459679 IC50 = 940 nM T66252 CKZ17B 71463121 IC50 = 8600 nM T66252 C4VKM3 71463122 IC50 = 8800 nM T66252 C7B8AO 71621488 IC50 = 12500 nM T66252 C8T2PW 71655265 IC50 = 1000 nM T66252 CVB75Q 71655394 IC50 = 650 nM T66252 CH4ZS0 71655395 IC50 > 100000 nM T66252 CW3JG7 71731241 IC50 > 100000 nM T66252 C3D4HJ 71731243 IC50 > 100000 nM T66252 CU6BC5 71731355 IC50 > 100000 nM T66252 C5TS9Y 71731356 IC50 > 100000 nM T66252 C5RTY9 71731357 IC50 > 100000 nM T66252 CD9F5X 71731476 IC50 > 100000 nM T66252 C3IO9H 71731477 IC50 > 100000 nM T66252 CVAD62 71731478 IC50 > 100000 nM T66252 C1ON0X 71731479 IC50 > 100000 nM T66252 CZYQ05 71731604 IC50 > 100000 nM T66252 C40YRO 71731605 IC50 > 100000 nM T66252 C9Q8MO 72164809 IC50 = 630 nM T66252 CL5X1Z 72164811 IC50 = 620 nM T66252 C7N8WB 72164813 IC50 = 1610 nM T66252 C2R0NV 72164815 IC50 = 450 nM T66252 C4JLM5 72164817 IC50 = 340 nM T66252 C6RQ9A 72164819 IC50 = 360 nM T66252 C38GWP 72164942 IC50 = 440 nM T66252 C4T0MY 72164944 IC50 = 280 nM T66252 C0T4UW 72164946 IC50 = 350 nM T66252 CLV02R 72164948 IC50 = 340 nM T66252 CHPN10 72164950 IC50 = 550 nM T66252 CI78FQ 72165082 IC50 = 310 nM T66252 CN0VU2 72165084 IC50 = 330 nM T66252 C84SYX 72165086 IC50 = 440 nM T66252 C1RQA3 72165088 IC50 = 260 nM T66252 CH51ZR 72165090 IC50 = 600 nM T66252 C65DFP 72697059 IC50 = 6500 nM T66252 CX07OC 72697060 IC50 = 2000 nM T66252 CZ56DO 72697061 IC50 = 4060 nM T66252 C1A2KX 72697062 IC50 = 20150 nM T66252 CS5U1F 72697063 IC50 = 8090 nM T66252 CA3HI1 72697064 IC50 = 2030 nM T66252 CCZJ47 72697206 IC50 = 1390 nM T66252 CWNZ91 72697207 IC50 = 8140 nM T66252 C6BWI4 72697208 IC50 = 11140 nM T66252 C9JA1Q 72697209 IC50 = 4720 nM T66252 CF6A8N 72697210 IC50 = 1950 nM T66252 CTMR03 72697211 IC50 = 9720 nM T66252 CP9NV5 72697212 IC50 = 15970 nM T66252 C1P8HS 72697352 IC50 = 22900 nM T66252 CC7G3M 72697353 IC50 = 9460 nM T66252 CXYO73 72697354 IC50 = 2030 nM T66252 CAXV78 72697355 IC50 = 19790 nM T66252 CGV09W 72697356 IC50 = 1390 nM T66252 CIF9D7 72697357 IC50 = 1760 nM T66252 CC8RA6 72697358 IC50 = 2867 nM T66252 C1EC7S 72697359 IC50 > 58000 nM T66252 C8CRO6 72697494 IC50 = 1290 nM T66252 C03NKY 72697495 IC50 = 2490 nM T66252 CP0MU3 72697496 IC50 = 9190 nM T66252 CI60AK 72697497 IC50 = 7740 nM T66252 CO19YK 72697498 IC50 = 5600 nM T66252 C47IGZ 72697499 IC50 = 3140 nM T66252 C65OPG 72697500 IC50 = 870 nM T66252 C3ZP7N 72697501 IC50 = 1000 nM T66252 C7EF8C 72697646 IC50 = 7360 nM T66252 C08IGP 72699737 IC50 > 100000 nM T66252 CAEF04 72707536 IC50 > 100000 nM T66252 C7ARW4 72707537 IC50 = 84500 nM T66252 CY0N9K 76311138 IC50 = 72400 nM T66252 CWK7M6 76311139 IC50 = 2000 nM T66252 CIP4R0 76314754 IC50 = 6800 nM T66252 C3HRA1 76314755 IC50 = 1300 nM T66252 C68JOX 76318341 IC50 = 10600 nM T66252 CET31O 76318342 IC50 = 1500 nM T66252 C9UGA3 76325642 IC50 > 288200 nM T66252 CNIP02 76325643 IC50 = 2600 nM T66252 C08DYM 76325644 IC50 = 2700 nM T66252 C3C7HE 76325645 IC50 = 7500 nM T66252 CW4M6E 76329221 IC50 = 5400 nM T66252 CH95ZJ 76336484 IC50 = 143600 nM T66252 CTXI04 86267501 IC50 > 10000 nM T66252 CO78UK 86267502 IC50 > 10000 nM T66252 CLG83C 86268944 IC50 > 10000 nM T66252 C31OGJ 86279928 IC50 > 10000 nM T66252 CIV7Y8 89668929 IC50 > 100000 nM T66252 CV0SF5 90664925 IC50 > 100000 nM T66252 CBQ38C 101879512 IC50 = 56720 nM T66252 CM7E4V 101887269 IC50 > 100000 nM T66252 C8EH0J 101887270 IC50 > 100000 nM T66252 CDT67J 101887271 IC50 > 100000 nM T66252 C4F2CS 101887272 IC50 > 100000 nM T66252 C58XWA 101887273 IC50 > 100000 nM T66252 C3Y9ET 101887274 IC50 > 100000 nM T66252 C1AF8C 101887275 IC50 > 100000 nM T66252 CH7QC5 101887276 IC50 > 100000 nM T66252 CO4FR2 101887277 IC50 > 100000 nM T66252 C9JEH0 101887278 IC50 > 100000 nM T66252 C52GIO 101887279 IC50 > 100000 nM T66252 CZ1G3O 118712516 IC50 > 100000 nM T66252 C8X4JA 118712517 IC50 > 100000 nM T66252 CC29AB 118712518 IC50 > 100000 nM T66252 CB09PD 118712519 IC50 > 100000 nM T66252 CD4U1X 118712520 IC50 > 100000 nM T66252 CU0V5J 118712521 IC50 > 100000 nM T66252 C03OUP 118712522 IC50 > 100000 nM T66252 CT2MZ8 118712764 IC50 = 170 nM T66252 C3W5RU 118712765 IC50 = 120 nM T66252 CKA1N5 118712766 IC50 = 30 nM T66252 C8M6ZW 118712767 IC50 = 620 nM T66252 CV5C6D 118712768 IC50 = 190 nM T66252 C2NSC7 118712769 IC50 = 140 nM T66252 CAR4W5 118712772 IC50 = 40 nM T66252 CRWT85 118712773 IC50 = 230 nM T66252 C4T2FY 118712775 IC50 = 330 nM T66252 C8IF4E 118712777 IC50 = 107660 nM T66252 CJ8EL0 118712778 IC50 = 22270 nM T66252 C07UOL 118712779 IC50 = 70460 nM T66252 C25HYG 118712780 IC50 = 21620 nM T66252 CD0HQ4 118712781 IC50 = 21960 nM T66252 C46TMQ 118712785 IC50 = 880 nM T66252 C5M3BX 118712788 IC50 = 5660 nM T66252 CK7HN4 118722408 IC50 = 15960 nM T66252 CK71WT 118722410 IC50 = 2180 nM T66252 CI74ZM 118722411 IC50 = 3300 nM T66252 CH1P7Y 118722412 IC50 = 1960 nM T66252 CL8TY5 118722413 IC50 = 6270 nM T66252 C8KUP0 118722416 IC50 = 320 nM T66252 COG4V6 118722421 IC50 = 5260 nM T66252 C7TEY3 122178433 IC50 > 10000 nM T66252 CN78TQ 122189864 IC50 > 100000 nM T66252 CNM82F 122189865 IC50 > 100000 nM T66252 C19GHJ 122189866 IC50 > 100000 nM T66252 C3U9KC 122189867 IC50 > 100000 nM T66252 CW5V3U 122189868 IC50 > 100000 nM T66252 CCG05R 122189869 IC50 > 100000 nM T66252 CI01PT 122189870 IC50 = 6300 nM T66252 C80EWF 122189871 IC50 > 100000 nM T66252 C3N7JC 122189872 IC50 > 100000 nM T66252 CG8O1J 122189873 IC50 > 100000 nM T66252 CK0US2 122189874 IC50 > 100000 nM T66252 C5V6NI 122189875 IC50 > 100000 nM T66252 CV7A9Y 122189876 IC50 > 100000 nM T66252 CH97SN 122189877 IC50 > 100000 nM T66252 CN86VR 122189878 IC50 > 100000 nM T66252 CZB49I 122189879 IC50 > 100000 nM T66252 CRM4Q8 135518358 IC50 > 100000 nM T66252 CMI5A6 135964368 IC50 = 56000 nM T66252 CO04QA 136177302 IC50 > 100000 nM T66252 C3SKH4 145948172 IC50 = 46000 nM T66252 CR9S6F 145958227 IC50 > 300000 nM T66252 CBL76R 145964231 IC50 > 100000 nM T66252 CF53NA 145964407 IC50 > 100000 nM T66252 CNMT16 145965136 IC50 > 100000 nM T66252 CP7VT2 145973710 IC50 > 100000 nM T66252 C9C4WU 145975568 IC50 > 100000 nM T66252 CWF4Y7 145977953 IC50 > 100000 nM T66252 CR3I9D 145978547 IC50 > 100000 nM T66252 CM6L4K 155510749 IC50 > 100000 nM T66252 C5ZQ7W 155511281 IC50 > 100000 nM T66252 CQA73O 155512586 IC50 > 100000 nM T66252 C57QZJ 155512836 IC50 > 100000 nM T66252 CX3U8Z 155515016 IC50 > 100000 nM T66252 C19ZCJ 155518265 IC50 > 100000 nM T66252 C8UOJ4 155518381 IC50 > 100000 nM T66252 CW0NI8 155519444 IC50 > 100000 nM T66252 C3I8AW 155520161 IC50 > 100000 nM T66252 C4AZ9V 155523785 IC50 > 100000 nM T66252 CTSA30 155526359 IC50 > 100000 nM T66252 CVD89H 155526728 IC50 > 100000 nM T66252 C5C4UV 155526759 IC50 > 100000 nM T66252 CAT3J0 155526949 IC50 > 100000 nM T66252 CLE9I0 155528648 IC50 > 100000 nM T66252 C8FHJ2 155529886 IC50 > 100000 nM T66252 CCX9H6 155530472 IC50 > 100000 nM T66252 CB6N4S 155531120 IC50 > 100000 nM T66252 CGV6C1 155531169 IC50 > 100000 nM T66252 CEOQ32 155531330 IC50 > 100000 nM T66252 CN04KW 155533304 IC50 > 100000 nM T66252 CG3RS6 155540249 IC50 > 100000 nM T66252 CJ67GL 155540375 IC50 > 100000 nM T66252 CY25EZ 155544299 IC50 > 100000 nM T66252 C8H3MJ 155544665 IC50 > 100000 nM T66252 CU17DA 155544967 IC50 > 100000 nM T66252 C62YMT 155545522 IC50 > 100000 nM T66252 CNA9X4 155548276 IC50 > 100000 nM T66252 CM9K4B 155548792 IC50 > 100000 nM T66252 CB1AF4 155549522 IC50 > 100000 nM T66252 CX9Y4B 155552378 IC50 > 100000 nM T66252 C1D5QZ 155554658 IC50 > 100000 nM T66252 C7KVR5 155559306 IC50 > 100000 nM T66252 C68CRH 155561682 IC50 > 100000 nM T66252 C48ETF 155565121 IC50 > 100000 nM T66252 CI5C6P 155568161 IC50 > 100000 nM T66252 CUQL05 155568269 IC50 > 100000 nM T66252 D03DNV 71655266 IC50 = 3400 nM T66252 D04CAR 10607286 Ki = 0.41 nM T66252 D07ALM 11232124 IC50 = 76600 nM T66252 D08NMS 46900258 Ki = 0.19 nM T66252 D0CP1J 56658139 IC50 = 53 nM T66252 D0L9XR 447256 IC50 = 11300 nM T66252 D0N1FU 6918465 IC50 = 6600 nM T66252 D0R5OE 44422449 IC50 = 6129 nM T66252 D0Y5IQ 44255320 IC50 = 10000 nM T64830 D02XIY 448601 IC50 = 22 nM T64830 D0TV0C 9941444 Ki = 0.1259 nM T64830 D06JFI 11251755 IC50 = 46 nM T64830 D0J8PI 158782 IC50 = 393 nM T64830 D09JXL 5311430 Ki = 12.59 nM T64830 D0Y2HR 2247 Ki = 4070 nM T64830 C6XYL5 6918011 Ki = 3.981 nM T64830 CHM63P 6918026 Ki = 5.012 nM T64830 CR0U6E 9827283 Ki > 10000 nM T64830 CA8UQ7 9848232 Ki > 10000 nM T64830 CW3TM5 9851998 Ki = 416 nM T64830 CTRI07 9852911 Ki = 3700 nM T64830 C9BJ3Q 9854636 IC50 = 633 nM T64830 CMLP16 9918828 Ki = 25 nM T64830 CG0U4Q 9937014 IC50 = 0.4 nM T64830 CF6TA4 9959983 IC50 > 100 nM T64830 C3Z5YJ 9963342 Ki = 0.3981 nM T64830 CIT57N 9985523 Ki = 5100 nM T64830 CL6G0Z 10094509 Ki = 1620 nM T64830 C9C7RK 10096510 Ki = 360 nM T64830 CFZN71 10166743 Ki = 691 nM T64830 CI21CK 10179247 Ki > 10000 nM T64830 C6DRE9 10210016 Ki = 2250 nM T64830 C4M9GN 10248767 Ki = 430 nM T64830 CSY5K2 10325243 Ki = 3000 nM T64830 CL87OB 10411795 Ki = 3650 nM T64830 CS96ON 10534086 IC50 = 30.3 nM T64830 CHZ9I8 10554930 Ki = 4000 nM T64830 CY3ZE9 10577746 IC50 = 87 nM T64830 C9C0HF 10580397 Ki = 1300 nM T64830 CU3DQ6 10630127 Ki = 48 nM T64830 C45JIZ 10699714 Ki = 3400 nM T64830 CG2UX4 10701257 IC50 = 2359 nM T64830 CP0F7C 10724811 IC50 = 3700 nM T64830 C3TMY5 10724880 IC50 = 152 nM T64830 CJM47E 10748701 IC50 = 208 nM T64830 CWF2N5 10748831 IC50 = 501 nM T64830 CLW4V6 10770814 Ki = 3900 nM T64830 CO56HI 10772403 IC50 = 1000 nM T64830 CGN0Z5 10772578 IC50 = 769 nM T64830 C3L4DH 10796238 IC50 = 123 nM T64830 C15QGO 10819673 IC50 = 1000 nM T64830 CFL71O 10843862 IC50 = 1176 nM T64830 C2PJ1O 10876898 Ki = 0.631 nM T64830 C6TVQ8 10964197 Ki = 0.3981 nM T64830 CXDG12 10996788 Ki = 0.1 nM T64830 C6AW0M 11112736 Ki = 3700 nM T64830 CK1RX4 11136828 Ki = 0.3162 nM T64830 CR1JP9 11147505 Ki = 3.162 nM T64830 C1I9EX 11159133 IC50 = 557 nM T64830 C7REL4 11170698 IC50 = 20.3 nM T64830 CIEM12 11170867 IC50 = 547 nM T64830 CW2JA8 11182381 IC50 = 17.5 nM T64830 CE3GC2 11205475 IC50 = 14 nM T64830 CXI32T 11205496 IC50 = 30 nM T64830 C2RNJ5 11205515 IC50 = 240 nM T64830 CUT8Z0 11240205 IC50 = 221 nM T64830 CK78SD 11240206 IC50 = 63 nM T64830 C67WXD 11274767 IC50 = 4.8 nM T64830 COK06N 11320738 IC50 = 147 nM T64830 C5D6AM 11332138 IC50 = 199 nM T64830 C5PAN4 11343811 IC50 = 110 nM T64830 CLQ53A 11355270 IC50 = 18 nM T64830 CQ0UC7 11378229 IC50 = 6 nM T64830 CC09ZU 11378299 IC50 = 692 nM T64830 CG7PT9 11389178 IC50 > 1000 nM T64830 CFJD72 11423410 IC50 = 51 nM T64830 C4S2HG 11434734 IC50 = 42 nM T64830 C6XHC3 11457491 IC50 = 1000 nM T64830 CJ5A9B 11457521 IC50 = 103 nM T64830 CMA8C7 11468709 IC50 > 1000 nM T64830 CG8A0J 11468887 IC50 = 24 nM T64830 CZ3N5J 11468916 IC50 = 7.6 nM T64830 CORY59 11480246 IC50 = 27 nM T64830 C63QMX 11535351 IC50 = 203 nM T64830 CF6K7M 11563877 IC50 = 1700 nM T64830 CS68YA 11642413 IC50 = 6000 nM T64830 CZHN61 11678313 IC50 = 50 nM T64830 CW65KY 11705763 Ki = 0.38 nM T64830 CN63YV 11787877 IC50 > 1000 nM T64830 CR6UF9 11788180 IC50 > 1000 nM T64830 CK4U8N 11804376 IC50 = 2741 nM T64830 C9XH7F 11815114 Ki = 0.2512 nM T64830 CRA01O 11845058 IC50 = 77 nM T64830 C8X3CL 11845059 IC50 = 539 nM T64830 CO3HT9 11847587 IC50 = 109 nM T64830 CAD8P9 11848624 Ki = 121 nM T64830 CM49QW 11848625 Ki = 199 nM T64830 CEBA46 11848626 Ki = 178 nM T64830 CCT5G7 11848677 Ki = 185 nM T64830 CMR10F 11848679 Ki = 13 nM T64830 C9QDX3 11848833 Ki = 31 nM T64830 CL6B5X 11848835 Ki = 8 nM T64830 CBV2X0 11963995 Ki = 15 nM T64830 CRIY45 12891521 Ki = 5000 nM T64830 C9P2IK 12891558 Ki > 10000 nM T64830 CW7I8U 13690207 IC50 = 0.77 nM T64830 C8OU7I 15429504 IC50 = 28 nM T64830 CEO3F0 15585102 IC50 = 27 nM T64830 C8IJ0O 15952316 Ki = 60 nM T64830 CC2YJ8 16062553 Ki = 23 nM T64830 C3H1RT 16062555 Ki = 18 nM T64830 C1LH5T 16062816 Ki = 3 nM T64830 C1GKF8 16130982 Ki = 0.46 nM T64830 C2TRA5 16144717 IC50 = 290 nM T64830 CW20OC 16144977 IC50 = 524 nM T64830 CS6A3Z 16145268 IC50 = 1247 nM T64830 CN3LS1 16145579 IC50 = 21.6 nM T64830 C72MUC 16146425 IC50 = 744 nM T64830 CD91IL 16148220 IC50 = 1837 nM T64830 C59OUC 16148481 Ki = 100 nM T64830 CJG1X9 16148596 Ki = 6.31 nM T64830 CNY09C 16148922 Ki = 100 nM T64830 CP0DC8 16149640 Ki = 0.3981 nM T64830 CDPC19 16149975 Ki = 0.631 nM T64830 C0SE6V 16150676 Ki = 0.1585 nM T64830 CSP6A9 16150915 Ki = 0.7943 nM T64830 C6N7SR 16151159 Ki = 79.43 nM T64830 C2B9IL 16151570 IC50 > 1000 nM T64830 CQM8J1 16151781 IC50 = 317 nM T64830 CM8UF7 16151826 IC50 > 1000 nM T64830 CJ7UT6 16151923 IC50 = 990 nM T64830 CIM03U 16152257 IC50 = 663 nM T64830 CU7X6V 16153077 IC50 = 393 nM T64830 CK4O1V 16153193 IC50 = 34 nM T64830 C16LMW 16153418 IC50 > 1000 nM T64830 CO0LG7 16154000 IC50 = 458 nM T64830 CX4RM8 16154096 IC50 = 19 nM T64830 COYU86 16156815 Ki = 79.43 nM T64830 CI3FW1 16157160 IC50 = 130 nM T64830 C7GN0S 16157479 Ki = 1.259 nM T64830 CQL5O0 16181427 IC50 > 1000 nM T64830 C2CUY9 16181428 IC50 > 1000 nM T64830 CUH8D7 16737812 IC50 = 318 nM T64830 C8QIT3 16737813 IC50 = 245 nM T64830 CNP36U 16737814 IC50 = 1.2 nM T64830 C7Q6JL 16738359 IC50 = 8 nM T64830 CUL5E0 24740295 Ki = 17 nM T64830 C0P6HM 24740408 Ki > 10000 nM T64830 CT1U3B 24740517 Ki > 10000 nM T64830 C0R7DJ 24740518 Ki = 6120 nM T64830 CIX0B4 24740519 Ki = 3950 nM T64830 C8PG7A 24740520 Ki = 1630 nM T64830 CY4RT7 24740521 Ki = 3950 nM T64830 CZL7D0 24740635 Ki = 1440 nM T64830 CH52FI 24740636 Ki = 1230 nM T64830 CD1H2Z 24740637 Ki = 683 nM T64830 CR2F4Q 24740638 Ki = 5128 nM T64830 C57RUG 24740639 Ki = 1789 nM T64830 CIB3C0 24740640 Ki = 149 nM T64830 CTX9A2 24740748 Ki = 326 nM T64830 CMC16R 24740749 Ki = 794 nM T64830 CJ9K1C 24740750 Ki = 66 nM T64830 CS6VO9 24740751 Ki = 83 nM T64830 CA4K0B 24740752 Ki = 23 nM T64830 C4N3AX 24740753 Ki = 293 nM T64830 COQU12 24740861 Ki = 487 nM T64830 CAD4S1 24740862 Ki = 194 nM T64830 C67YVI 24740863 Ki = 113 nM T64830 CO0IF5 24740864 Ki = 37 nM T64830 CAX2F4 24740865 Ki = 524 nM T64830 C6F1RZ 24777672 IC50 = 206 nM T64830 C5GZO7 24858018 IC50 = 28 nM T64830 CV1U7H 24858920 IC50 = 9.5 nM T64830 C0UB7K 24859055 IC50 = 8.7 nM T64830 CQCW58 24859056 IC50 = 26 nM T64830 CT6J2A 24859195 IC50 = 9.1 nM T64830 CUDV69 24859196 IC50 = 11 nM T64830 C45NYA 24859341 IC50 = 7.4 nM T64830 C4AB6I 24859342 IC50 = 46 nM T64830 CH50QU 24859494 IC50 = 9 nM T64830 C8L2KJ 24859495 IC50 = 82 nM T64830 CDS6W5 24859645 IC50 = 50 nM T64830 CHF20D 24859646 IC50 = 17 nM T64830 CKH2R4 24859787 IC50 = 51 nM T64830 CT1BM6 24859788 IC50 = 50 nM T64830 C2IKX3 24859919 IC50 = 50 nM T64830 C5OQ2X 24859920 IC50 = 107 nM T64830 CSZ73L 24860057 IC50 = 60 nM T64830 C36ZHQ 24860058 IC50 = 21 nM T64830 CVL48C 24860201 IC50 = 57 nM T64830 C20ZFS 24860202 IC50 = 90 nM T64830 CI8BZ6 24936235 Ki > 100000 nM T64830 C07OMT 25122324 IC50 = 83 nM T64830 CHKC79 25187396 IC50 = 5 nM T64830 C4YXJ1 25187398 IC50 = 3.4 nM T64830 CO9PI7 25187400 IC50 = 1.8 nM T64830 C8C9PL 25187679 IC50 = 3.7 nM T64830 C9ECD8 25187681 IC50 = 16 nM T64830 C43OES 25187683 IC50 = 8.8 nM T64830 CNTB73 25187685 IC50 = 1.4 nM T64830 C1IUQ2 25187953 IC50 = 8 nM T64830 CQ3F8L 25187955 IC50 = 2.9 nM T64830 CS2ZV1 25188218 IC50 = 50 nM T64830 CLI2U1 25188220 IC50 = 3.2 nM T64830 CNDU95 25188496 IC50 = 13 nM T64830 C7KF8N 25188776 IC50 = 25 nM T64830 CCHN50 25188780 IC50 = 0.56 nM T64830 C3T8DA 25189052 IC50 = 0.86 nM T64830 CI21ED 25189054 IC50 = 3.5 nM T64830 C97LHK 25189325 IC50 = 0.6 nM T64830 CEG4J0 25189327 IC50 = 3.5 nM T64830 CSQH26 42637069 IC50 > 1000 nM T64830 CJ1S9K 42637136 IC50 > 1000 nM T64830 C3NYM8 42637137 IC50 > 1000 nM T64830 CJ47CL 42637210 IC50 > 1000 nM T64830 CR3A8Q 42637283 IC50 > 1000 nM T64830 CENZ47 42637363 IC50 > 1000 nM T64830 CX0JC7 42637503 IC50 > 1000 nM T64830 C90LHS 42637563 IC50 > 1000 nM T64830 C80WBK 42637632 IC50 > 1000 nM T64830 CR49YE 42637984 IC50 > 1000 nM T64830 CEFO24 42638065 IC50 > 1000 nM T64830 CF5JK4 42638066 IC50 > 1000 nM T64830 CHY04A 44290718 IC50 = 2.8 nM T64830 C16BKW 44290734 IC50 = 1 nM T64830 CW76YB 44290735 IC50 = 7.8 nM T64830 CA6IS7 44290766 IC50 = 1.3 nM T64830 C6BZ1J 44298104 Ki = 524 nM T64830 CCXL10 44298113 Ki = 139 nM T64830 CYW8O0 44298130 Ki = 204 nM T64830 CB9JK1 44298131 Ki = 70 nM T64830 CJ5WL8 44298155 Ki = 304 nM T64830 CHL57J 44298156 Ki = 1860 nM T64830 CP61LB 44298165 Ki = 461 nM T64830 CM0B6J 44298166 Ki = 725 nM T64830 C8XZR7 44298169 Ki = 376 nM T64830 C0DPX7 44298171 Ki = 382 nM T64830 C62OEU 44298177 Ki = 748 nM T64830 CS9JW8 44298178 Ki = 694 nM T64830 C20MBI 44298179 Ki = 173 nM T64830 C3QBP0 44298188 Ki = 960 nM T64830 C1R3QD 44298189 Ki = 48 nM T64830 C5RJ7U 44298195 Ki = 369 nM T64830 C8N3EJ 44298197 Ki = 87 nM T64830 CZU05A 44298214 Ki = 689 nM T64830 CQUS98 44298218 Ki = 972 nM T64830 COTK07 44298219 Ki = 1580 nM T64830 CAJO07 44298231 Ki = 968 nM T64830 C9S4IX 44298232 Ki = 814 nM T64830 CB1A3K 44298235 Ki = 847 nM T64830 C2TQ1V 44298248 Ki = 926 nM T64830 C3WFV5 44298250 Ki = 66 nM T64830 CVW19Y 44298328 Ki = 1380 nM T64830 CT94HY 44298329 Ki = 918 nM T64830 CL4F1V 44298378 Ki = 110 nM T64830 CMO1Q9 44298441 Ki = 140 nM T64830 C8Y9ZP 44298443 Ki = 240 nM T64830 CUSR45 44298468 Ki = 468 nM T64830 C8EN2H 44298469 Ki = 734 nM T64830 CWE7Q0 44298482 IC50 > 10000 nM T64830 CF69PL 44298522 Ki = 287 nM T64830 CRQJ98 44308836 Ki = 5017 nM T64830 CRFM02 44308969 Ki = 4470 nM T64830 C40MJU 44308970 Ki = 2.32 nM T64830 C9KR7Q 44309052 Ki = 3316 nM T64830 C4YG1S 44311590 IC50 > 10000 nM T64830 CY0OV9 44311591 IC50 = 190 nM T64830 C29GQB 44311601 IC50 = 5 nM T64830 CC8DS0 44311602 IC50 > 10000 nM T64830 C5KST2 44311690 IC50 > 1000 nM T64830 C6N4MH 44311691 IC50 > 1000 nM T64830 CIR4G6 44311695 IC50 > 1000 nM T64830 CTG6X5 44311696 IC50 > 1000 nM T64830 C7Y8SF 44311697 IC50 > 1000 nM T64830 CK52MY 44311702 IC50 > 10000 nM T64830 CX39CV 44311703 IC50 > 1000 nM T64830 C5RM2A 44311730 IC50 > 1000 nM T64830 CBG70T 44311731 IC50 > 1000 nM T64830 CQH20F 44311765 IC50 > 10000 nM T64830 CZG4K6 44311836 IC50 > 1000 nM T64830 CWNP79 44311837 IC50 > 1000 nM T64830 CEMH98 44311848 IC50 = 4.92 nM T64830 CWSF38 44311868 IC50 > 10000 nM T64830 C2T0YP 44311869 IC50 > 1000 nM T64830 C1ONB3 44311870 IC50 = 385 nM T64830 C1LQN0 44311889 IC50 = 4.17 nM T64830 C1GY0F 44311912 IC50 > 1000 nM T64830 C14DIH 44311913 IC50 > 10000 nM T64830 C1X4TI 44311914 IC50 = 45.7 nM T64830 C64WAE 44311958 IC50 > 1000 nM T64830 CFT90E 44311959 IC50 > 10000 nM T64830 C3PQD0 44311960 IC50 > 10000 nM T64830 C3WFS2 44311993 IC50 = 10.95 nM T64830 CS7PB4 44312258 IC50 > 10000 nM T64830 C2LZI6 44312330 IC50 = 0.77 nM T64830 C5PE1D 44325273 IC50 = 41 nM T64830 C1P0QV 44332931 Ki > 10000 nM T64830 CQ2ID4 44345936 IC50 = 398.11 nM T64830 C0U1IB 44345981 IC50 = 1412.54 nM T64830 C8JMF4 44346082 IC50 = 316.23 nM T64830 C7I9RK 44346098 IC50 = 316.23 nM T64830 C2Z9BG 44346106 IC50 = 501.19 nM T64830 CAG1Z4 44354386 Ki > 10000 nM T64830 C3QZH1 44354398 Ki = 2858 nM T64830 C3KS5A 44354415 Ki = 333 nM T64830 CHP41F 44363816 Ki = 284 nM T64830 CH2DN4 44367916 IC50 > 10000 nM T64830 CM9YQ0 44367953 IC50 > 1000 nM T64830 C5W4YL 44368019 IC50 > 1000 nM T64830 CO6ZJ9 44368020 IC50 > 1000 nM T64830 CQ5T1D 44368043 IC50 = 127 nM T64830 C1SWO5 44368044 IC50 > 1000 nM T64830 C29EZK 44368080 IC50 = 23 nM T64830 C9ZW6U 44368093 IC50 = 700 nM T64830 C71URM 44368094 IC50 = 47 nM T64830 CC1ZP9 44368109 IC50 > 10000 nM T64830 CQ7OP1 44368112 IC50 = 101 nM T64830 C0EW4I 44368117 IC50 = 152 nM T64830 C6TNZ9 44368144 IC50 > 1000 nM T64830 C53IAG 44368153 IC50 = 27 nM T64830 CKU8J7 44368156 IC50 = 14 nM T64830 CR12GB 44368157 IC50 = 46 nM T64830 C50DMO 44368226 IC50 > 10000 nM T64830 CN31HS 44368398 IC50 = 34 nM T64830 C2RC0P 44368406 IC50 = 211 nM T64830 CB1HC8 44368422 IC50 > 1000 nM T64830 C27DLY 44368489 IC50 > 1000 nM T64830 CWHK38 44377332 Ki > 10000 nM T64830 CVH1O7 44377366 Ki > 5000 nM T64830 CRC2N1 44377555 Ki = 600 nM T64830 CS1WT5 44377591 Ki = 2300 nM T64830 C3LUY8 44377623 Ki = 540 nM T64830 CQD0P4 44377645 Ki > 5000 nM T64830 CWNF42 44385504 Ki = 1130 nM T64830 CAFD79 44385508 Ki > 10000 nM T64830 CHY14B 44385591 Ki > 10000 nM T64830 CJQI19 44385652 Ki = 2360 nM T64830 CG12HD 44385712 Ki = 1190 nM T64830 C8MU5C 44385757 Ki = 1870 nM T64830 C0LRT9 44386389 Ki = 2120 nM T64830 C1EVK8 44387399 Ki > 1000 nM T64830 C6U9VC 44388027 IC50 > 1000 nM T64830 C2IW5J 44388028 IC50 > 1000 nM T64830 C27ANT 44388029 IC50 > 1000 nM T64830 CHQK20 44388035 IC50 > 1000 nM T64830 CI9XS1 44388036 IC50 > 1000 nM T64830 CD4BX6 44388037 IC50 > 1000 nM T64830 CDS08Z 44388038 IC50 > 1000 nM T64830 CZA03Y 44388040 IC50 > 1000 nM T64830 C21WBR 44388043 IC50 > 1000 nM T64830 C7VK6B 44388052 IC50 > 1000 nM T64830 CT93BI 44388060 IC50 > 1000 nM T64830 C4E5VS 44388061 IC50 > 1000 nM T64830 C7P5RO 44388066 IC50 > 1000 nM T64830 C7T8IY 44388069 IC50 > 1000 nM T64830 C2TWO3 44388070 IC50 > 1000 nM T64830 CDBE87 44388075 IC50 > 1000 nM T64830 C25GWK 44388078 IC50 > 1000 nM T64830 CT93LV 44388079 IC50 > 1000 nM T64830 CX54SC 44388083 IC50 = 682 nM T64830 C2C0RU 44388084 IC50 > 1000 nM T64830 C5SMA2 44388085 IC50 > 1000 nM T64830 C26OCG 44388086 IC50 = 803 nM T64830 C8SR2O 44388087 IC50 > 1000 nM T64830 CHL5T1 44388088 IC50 > 1000 nM T64830 C4VNC2 44388089 IC50 > 1000 nM T64830 C1IH3T 44388090 IC50 > 1000 nM T64830 CNC91I 44388093 IC50 > 1000 nM T64830 CN45OF 44388095 IC50 > 1000 nM T64830 C82HJL 44388104 IC50 > 1000 nM T64830 CV6T2H 44388105 IC50 > 1000 nM T64830 CLC0N2 44388106 IC50 > 1000 nM T64830 C0VO1K 44388107 IC50 > 1000 nM T64830 CM5O3B 44388108 IC50 > 1000 nM T64830 CAF02P 44388109 IC50 > 1000 nM T64830 C23XBM 44388110 IC50 > 1000 nM T64830 CPX74G 44388112 IC50 > 1000 nM T64830 CG9SA3 44388114 IC50 > 1000 nM T64830 C2C4MH 44388116 IC50 > 1000 nM T64830 CW1EL5 44388118 IC50 > 1000 nM T64830 CN0K3V 44388119 IC50 > 1000 nM T64830 CE8DH4 44388120 IC50 > 1000 nM T64830 C1A0OY 44388121 IC50 > 1000 nM T64830 CS53NP 44388122 IC50 > 1000 nM T64830 CX67WG 44388123 IC50 > 1000 nM T64830 CB50EK 44388124 IC50 > 1000 nM T64830 C9SN1X 44388132 IC50 > 1000 nM T64830 C6W4YT 44388133 IC50 > 1000 nM T64830 CMTN20 44388134 IC50 > 1000 nM T64830 CAK42W 44388135 IC50 > 1000 nM T64830 CTW48B 44388136 IC50 > 1000 nM T64830 C4P1AS 44388137 IC50 > 1000 nM T64830 CEAZ82 44388138 IC50 > 1000 nM T64830 CZ2K1I 44397385 Ki = 56 nM T64830 C1KMT8 44397389 Ki = 1.7 nM T64830 C83JNK 44397472 Ki = 7.8 nM T64830 CE6U2K 44397620 Ki = 10 nM T64830 CM1W3L 44397628 Ki = 27 nM T64830 CN6Z8C 44397648 Ki = 8.4 nM T64830 CRW0M6 44397706 Ki = 2.1 nM T64830 CL7GX3 44397725 Ki = 70 nM T64830 C30MBR 44397747 Ki = 51 nM T64830 CQ0M7K 44397788 Ki = 64 nM T64830 C3MG9D 44397815 Ki = 1300 nM T64830 CK19EU 44397834 Ki = 66 nM T64830 C0OZB8 44397835 Ki = 2.3 nM T64830 C7X2VS 44397875 Ki = 26 nM T64830 C9DMA7 44397907 Ki = 58 nM T64830 CAD5S1 44397924 Ki = 9.3 nM T64830 C20TXF 44397990 Ki = 410 nM T64830 CM1R8X 44400000 IC50 = 114 nM T64830 CP89CS 44400135 IC50 = 377 nM T64830 CV4PO0 44403186 IC50 = 14 nM T64830 C8MEP3 44403194 IC50 = 1 nM T64830 C9B3AP 44403195 IC50 = 0.65 nM T64830 C29GND 44403204 IC50 = 54 nM T64830 CM3KG6 44403206 IC50 = 2.9 nM T64830 C0DG2C 44403217 IC50 = 10 nM T64830 C9MBD4 44403227 IC50 = 3.4 nM T64830 CLH53T 44403242 IC50 = 74 nM T64830 CIEM04 44403248 IC50 = 30 nM T64830 CX87AN 44435319 Ki > 10000 nM T64830 CCYM90 44435539 Ki = 1100 nM T64830 C7SA5B 44435540 Ki = 120 nM T64830 C8WID5 44435541 Ki = 20 nM T64830 C7UN0V 44435542 Ki = 40 nM T64830 C1BY2P 44444935 IC50 = 28 nM T64830 CH17TI 44560858 IC50 = 276 nM T64830 C2AZY7 44560859 IC50 > 1000 nM T64830 C2I8NB 44560860 IC50 > 1000 nM T64830 C4XRT0 44560861 IC50 > 1000 nM T64830 C21TZI 44560862 IC50 > 1000 nM T64830 C2YM5N 44560863 IC50 > 1000 nM T64830 CS39FB 44560864 Ki = 48 nM T64830 CU3FD2 44560865 Ki = 50 nM T64830 C8IKU1 44560866 IC50 = 442 nM T64830 CTQ83Z 44560867 IC50 = 728 nM T64830 CQC29N 44560868 IC50 = 657 nM T64830 C47MDA 44560869 IC50 = 149 nM T64830 CHAJ41 44560870 IC50 = 111 nM T64830 CT0A9U 44560871 IC50 > 1000 nM T64830 CM0T9R 44560872 IC50 > 1000 nM T64830 CO2J6R 44560873 IC50 = 895 nM T64830 CKQD64 44560874 IC50 = 461 nM T64830 CEK26Y 44560875 IC50 = 247 nM T64830 CBL1P7 44560876 IC50 = 320 nM T64830 CY47DM 44560877 IC50 = 191 nM T64830 C5OZD1 44560878 IC50 = 560 nM T64830 CFT47C 44560898 IC50 = 810 nM T64830 CAO7R0 44560899 IC50 = 313 nM T64830 C80ZCF 44560900 IC50 = 426 nM T64830 CATH94 44560901 IC50 = 94 nM T64830 C2AXG6 44560902 IC50 = 618 nM T64830 COQ9W7 44560903 IC50 > 1000 nM T64830 CLZ23V 44560904 IC50 > 1000 nM T64830 C0OKG2 44560905 IC50 > 1000 nM T64830 CPIW17 44560906 IC50 > 1000 nM T64830 CFR3Y5 44560907 IC50 > 1000 nM T64830 CS85LR 44560908 IC50 > 1000 nM T64830 C27GAF 44569760 IC50 = 12 nM T64830 CWDP17 44569804 IC50 = 0.3 nM T64830 C6K1FI 44577218 IC50 > 1000 nM T64830 CAJ15T 44577219 IC50 = 109 nM T64830 CQD56E 44577220 IC50 = 218 nM T64830 CV18IC 44577221 IC50 = 199 nM T64830 CLJD09 45102042 IC50 = 180 nM T64830 C63YJS 45139239 IC50 = 263 nM T64830 C63XPN 45267999 IC50 > 1000 nM T64830 CF09UA 45268875 IC50 > 1000 nM T64830 C2PNH4 45272264 IC50 > 1000 nM T64830 CFL9K7 45273129 IC50 = 218 nM T64830 C9Z4MR 45273130 IC50 > 1000 nM T64830 C4RGN0 45273131 IC50 = 9.9 nM T64830 CH18QA 46882131 Ki > 1000 nM T64830 CBZ3T9 46882132 Ki > 1000 nM T64830 C6KBJ2 46882133 Ki = 182 nM T64830 CNL16U 46882180 Ki = 252 nM T64830 CCX75M 46882181 Ki = 205 nM T64830 C2BOJ6 46882182 Ki = 52 nM T64830 C9ASC1 46882224 Ki = 55 nM T64830 CB38SE 46882225 Ki = 252 nM T64830 CP2N1U 46882226 Ki = 239 nM T64830 CJ3Q6B 46882227 Ki = 175 nM T64830 CRYQ47 46882445 Ki = 330 nM T64830 CRZ1B0 46882446 Ki > 1000 nM T64830 CNEZ46 46882447 Ki > 1000 nM T64830 C8D1OR 46882448 Ki > 1000 nM T64830 CZ0G2R 46882449 Ki > 1000 nM T64830 CR37UF 46882513 Ki > 1000 nM T64830 CF3L8U 46882514 Ki > 1000 nM T64830 C91WKZ 46882515 Ki > 1000 nM T64830 CX21JH 46882516 Ki = 361 nM T64830 CBJ92C 46882517 Ki = 309 nM T64830 C8N3KX 46882577 Ki = 194 nM T64830 CAH31I 46882578 Ki = 196 nM T64830 CD2NL0 46882579 Ki = 252 nM T64830 C9B0DF 46882620 Ki = 354 nM T64830 CJ8I4L 46882621 Ki = 357 nM T64830 C2YMA7 46882622 Ki = 226 nM T64830 CD0VH7 46882664 Ki = 343 nM T64830 C50YRJ 46882665 Ki = 633 nM T64830 CXFV62 46882666 Ki = 720 nM T64830 CR07WV 46882667 Ki > 1000 nM T64830 CF1HC7 46882668 Ki > 1000 nM T64830 CVIU56 46882708 Ki = 371 nM T64830 C8S4LN 46882709 Ki > 1000 nM T64830 CJ7GM9 46882746 Ki = 472 nM T64830 C6OM5H 46882789 Ki = 524 nM T64830 C5MV8K 46882790 Ki = 537 nM T64830 C6RD3V 46882791 Ki > 1000 nM T64830 C1WUF9 46882831 Ki = 33 nM T64830 C5LM3W 46882832 Ki = 156 nM T64830 CU1D6I 46902023 IC50 = 200 nM T64830 CZ46AH 46911015 IC50 = 3.1 nM T64830 CS8UX3 46911065 Ki = 18 nM T64830 CBF63L 49800498 IC50 = 1.1 nM T64830 C92UJY 49862886 Ki = 21 nM T64830 CX20EB 49862887 Ki = 19 nM T64830 C6O7TC 49862888 Ki = 4.9 nM T64830 C8B7ZO 49862889 Ki = 11 nM T64830 C0OAZ3 49862903 Ki = 436 nM T64830 C6Y7MJ 49862904 Ki = 11 nM T64830 C3A4QC 49862905 Ki = 4 nM T64830 CS9EY0 49862906 Ki = 4.4 nM T64830 CHF82N 49862928 Ki = 2.4 nM T64830 CE5R2Y 49862929 Ki = 7.1 nM T64830 CYL0N6 49862930 Ki = 6.3 nM T64830 CQN63O 49862931 Ki = 6.9 nM T64830 C79TRO 49862959 Ki = 7.9 nM T64830 C4XGC1 49862960 Ki = 5.4 nM T64830 C3UO2Y 49862961 Ki = 2.5 nM T64830 C7Y1FH 49862962 Ki = 6.7 nM T64830 C2K4LR 49862994 Ki = 18 nM T64830 C2VFO3 49862995 Ki = 637 nM T64830 CM7GK6 49862996 Ki = 22 nM T64830 CUM01E 49863042 Ki = 25 nM T64830 CLR0I7 49863043 Ki = 22 nM T64830 C14YCO 49863044 Ki = 9.3 nM T64830 CUXZ59 49863045 Ki > 1000 nM T64830 C84ZTC 49865341 IC50 = 28 nM T64830 C3VZ4U 49865342 IC50 = 29 nM T64830 CGYR09 49865343 IC50 = 12.3 nM T64830 C35WID 49865344 IC50 = 16.5 nM T64830 C0RK7G 49865345 IC50 = 418 nM T64830 C4YLM7 49865346 IC50 = 161 nM T64830 CZ4RI1 49865347 IC50 = 4.9 nM T64830 CQJP15 51003591 Ki = 5000 nM T64830 C9SNL1 52941607 IC50 = 200 nM T64830 CICK49 52944903 IC50 = 160 nM T64830 C3B8NF 52944904 IC50 = 160 nM T64830 CA78RK 52948576 IC50 = 70 nM T64830 CK4T3P 52948577 IC50 = 100 nM T64830 C40ZRY 52948630 IC50 = 70 nM T64830 C3R0CY 52948856 IC50 = 200 nM T64830 CED3O6 53473658 IC50 = 556 nM T64830 CE7J0U 53473659 IC50 = 41 nM T64830 CY0G2K 53473744 IC50 = 69 nM T64830 CBQG96 53473824 IC50 = 2.4 nM T64830 CW53YV 53473917 IC50 > 1000 nM T64830 C87SME 53474004 IC50 > 1000 nM T64830 C7EO1Z 53474005 IC50 > 1000 nM T64830 CY3M2A 53474090 IC50 > 1000 nM T64830 CM58UZ 56651206 IC50 = 3000 nM T64830 COBQ28 56651207 Ki = 1100 nM T64830 C9JHI4 56664813 Ki = 1.4 nM T64830 CU7SD5 56847878 IC50 = 0.8 nM T64830 C91BAH 56848075 IC50 = 1.1 nM T64830 C8ZW3O 56927659 IC50 = 533 nM T64830 CHK8T1 56945132 Ki > 10000 nM T64830 C73XBL 57384077 IC50 > 1000 nM T64830 C3KC9Z 57398462 IC50 = 2.9 nM T64830 C73HAD 66765125 IC50 = 1.5 nM T64830 C8AZH3 66765321 IC50 = 1.2 nM T64830 COE38P 66766052 IC50 = 0.3 nM T64830 CNPZ52 68093096 IC50 = 7.9 nM T64830 CDO5A6 68093280 IC50 = 0.8 nM T64830 C0DEM2 68254010 IC50 = 2.5 nM T64830 CTVI05 70683416 IC50 = 279 nM T64830 CV42WQ 70689221 IC50 = 220 nM T64830 C3P0AN 70689413 IC50 = 126 nM T64830 CP58HL 70689414 IC50 = 53 nM T64830 CB14OW 70689415 IC50 = 196 nM T64830 CNZC97 70689723 IC50 = 181 nM T64830 C2WQM9 70691295 IC50 > 1000 nM T64830 C5E8MY 70693613 IC50 = 137 nM T64830 C3TZ9U 70695246 IC50 = 302 nM T64830 C34XGS 70695722 IC50 = 76 nM T64830 CIPF50 70695723 IC50 = 247 nM T64830 CF08XL 71458043 Ki = 1200 nM T64830 CU82HG 71460000 IC50 > 1000 nM T64830 CPC69G 71461645 Ki = 790 nM T64830 CLAV92 71461684 IC50 > 1000 nM T64830 C1NZU3 71461685 IC50 > 10000 nM T64830 CFKH42 71717904 IC50 = 302 nM T64830 CGDO59 72947672 Ki = 0.2 nM T64830 CIO28F 73345407 Ki = 5.98 nM T64830 CMN6X8 73345525 IC50 > 1000 nM T64830 C70XZC 73345528 IC50 = 9 nM T64830 CXGJ67 73345700 IC50 = 65 nM T64830 CV23JS 73345701 IC50 = 521 nM T64830 C81UME 73345740 Ki = 1400 nM T64830 CX5VM1 73346900 IC50 > 10000 nM T64830 CA3MU5 73346903 IC50 = 16.7 nM T64830 C62NFY 73346927 Ki = 161 nM T64830 CK64MX 73346930 Ki = 766 nM T64830 C15CAN 73346972 Ki = 100.7 nM T64830 CD09FU 73347225 Ki = 153 nM T64830 CI4L6W 73347226 Ki = 469 nM T64830 CGM61R 73348311 Ki > 10000 nM T64830 CN1FD2 73348312 Ki > 10000 nM T64830 C01GIQ 73348427 Ki = 106 nM T64830 C7Y9ZT 73348428 Ki = 1000 nM T64830 CFLT50 73348719 IC50 = 91 nM T64830 C75NBQ 73348741 Ki = 631 nM T64830 C5MNX3 73348742 Ki = 2250 nM T64830 CL94MY 73350006 Ki = 101 nM T64830 C0N6XK 73350010 Ki = 40.1 nM T64830 CTV30F 73350011 Ki = 93 nM T64830 CF2AK4 73350012 Ki = 313 nM T64830 CK9CS4 73351516 Ki = 112 nM T64830 CNY13O 73351517 Ki = 176 nM T64830 CUN6L1 73351622 IC50 = 34 nM T64830 CC98JE 73351624 IC50 = 13 nM T64830 CWUH52 73351718 Ki = 45.5 nM T64830 CS9I4W 73351829 Ki = 535 nM T64830 CF70XH 73351873 IC50 > 1000 nM T64830 CFB54J 73352985 Ki = 140 nM T64830 CKFV85 73353009 Ki = 87 nM T64830 CC45AV 73353272 IC50 = 50 nM T64830 C41OCY 73353278 IC50 = 4.5 nM T64830 CW54CU 73353340 IC50 > 1000 nM T64830 CL7DT2 73354494 Ki = 1000 nM T64830 CA48EL 73354535 Ki = 33.5 nM T64830 CFK7Z3 73354633 IC50 = 668 nM T64830 C1UYL2 73354783 IC50 = 10.8 nM T64830 CG1CX0 73354798 IC50 = 18.2 nM T64830 CIVZ67 73354818 Ki = 520 nM T64830 CGCE64 73354819 Ki = 260 nM T64830 C1Y0CI 73356066 Ki = 1000 nM T64830 C52JAS 73356068 Ki = 88.5 nM T64830 CN5LG8 73356069 Ki = 1000 nM T64830 C9GKV2 73356181 IC50 = 397 nM T64830 C7XFB6 73356331 IC50 = 1.2 nM T64830 CI02SE 73356366 Ki = 140 nM T64830 CW8L6C 76310862 IC50 > 1000 nM T64830 CHV6K7 76314485 IC50 = 37 nM T64830 C0PR3Y 76314486 IC50 > 1000 nM T64830 C94BWD 76314487 IC50 = 25 nM T64830 C25XKO 76314488 IC50 = 16 nM T64830 CS54IV 76321777 IC50 = 50 nM T64830 C94OAT 76321778 IC50 = 58 nM T64830 CU1IR8 76325402 IC50 = 12 nM T64830 C17TRJ 78210294 IC50 = 6.2 nM T64830 CL09JQ 86279005 IC50 > 10000 nM T64830 C3JOS4 86292350 Ki > 9853 nM T64830 CVLE34 86293506 Ki > 9850 nM T64830 C15VTO 86294248 Ki > 9855 nM T64830 C64ALX 86299160 IC50 = 14 nM T64830 CP8X3E 89573118 IC50 = 2.1 nM T64830 CHYQ79 89573250 IC50 = 30 nM T64830 CO4I9D 89573308 IC50 = 3.2 nM T64830 CP4GJ3 89573310 IC50 = 5.7 nM T64830 CVI32M 89573420 IC50 = 0.4 nM T64830 CV3CZ7 89573523 IC50 = 0.4 nM T64830 CW4M0U 89573623 IC50 = 0.2 nM T64830 CV09DC 89583150 IC50 = 1.2 nM T64830 C47HED 89583208 IC50 = 0.4 nM T64830 C2GF8T 90423008 IC50 = 14 nM T64830 CJY3P0 90423921 IC50 = 9.6 nM T64830 CY6IE5 90423996 IC50 = 2.6 nM T64830 CI58FM 90663867 IC50 = 64 nM T64830 CK62FO 90663868 IC50 = 75 nM T64830 C7AFD4 90663869 IC50 = 413 nM T64830 C94XTF 90663872 IC50 = 110 nM T64830 CA7W0U 90663873 IC50 = 210 nM T64830 C4EG8T 90663874 IC50 = 327 nM T64830 CW21UO 90663875 IC50 = 310 nM T64830 C7Q4PD 90665458 Ki = 9500 nM T64830 CR43ZL 90665459 Ki = 28000 nM T64830 CLK7C3 90665460 Ki = 2100 nM T64830 CZ0UC6 90665461 Ki = 1700 nM T64830 C0IBJ6 90665462 Ki = 13200 nM T64830 CPX0C9 90665463 Ki = 11000 nM T64830 C3UVC8 91936728 IC50 = 73 nM T64830 CT3UP7 91936729 IC50 = 187 nM T64830 C1BW9G 101884861 Ki = 34000 nM T64830 CD2E4L 101941290 IC50 = 1000 nM T64830 C9KB3W 117711399 Ki > 9860 nM T64830 CTH52C 118718416 Ki = 1 nM T64830 CKQ4P6 118718462 IC50 = 347 nM T64830 C1Z7UJ 118718463 Ki < 1000 nM T64830 CPYA80 118718465 IC50 = 3356 nM T64830 CR61UD 118718466 IC50 = 1060 nM T64830 CW64XN 118718500 IC50 = 2032 nM T64830 CB4D5T 118718501 IC50 = 101 nM T64830 CW5HG2 118718502 IC50 = 1000 nM T64830 CC36KP 118718503 IC50 = 1000 nM T64830 C7FIQ1 118718504 IC50 = 1834 nM T64830 CNBY57 118718505 IC50 = 1484 nM T64830 CPY4Q5 118718506 IC50 = 529 nM T64830 CO13JR 118718507 IC50 = 470 nM T64830 CLFJ60 118718508 IC50 = 243 nM T64830 C13YUH 118718509 IC50 = 221 nM T64830 CP2O7U 118718510 IC50 = 178 nM T64830 CLDZ63 118718511 IC50 = 1959 nM T64830 CYQ7X2 118718854 IC50 = 460 nM T64830 CA6C4T 118719101 IC50 = 84 nM T64830 CDZ3H4 118719196 IC50 = 342 nM T64830 CQRO32 118719197 IC50 = 629 nM T64830 CGXH91 118719198 IC50 = 247 nM T64830 C1QJX7 118719199 IC50 = 50 nM T64830 C0GLC8 118719200 IC50 > 1000 nM T64830 C40NGQ 118719201 IC50 > 1000 nM T64830 CK2W9T 118719202 IC50 = 768 nM T64830 CW4AT0 118719275 IC50 > 1000 nM T64830 C5VWI1 118719303 IC50 = 358 nM T64830 CE8JW7 118897585 IC50 = 5.1 nM T64830 CT4S5C 118897590 IC50 = 18 nM T64830 CVI2N7 118897591 IC50 = 2.1 nM T64830 C9FW6P 118897690 IC50 = 30 nM T64830 CGRV31 118897691 IC50 = 6.1 nM T64830 CXW8A6 118897700 IC50 = 5.7 nM T64830 C9FJD3 118897882 IC50 = 3.9 nM T64830 C1X8US 118897967 IC50 = 4.6 nM T64830 CH6IT9 118897987 IC50 = 7.3 nM T64830 C5AJ7E 118898094 IC50 = 58 nM T64830 C7HA5C 118898105 IC50 = 6.7 nM T64830 CHUW06 118898153 IC50 = 6.1 nM T64830 CH6E5G 118963835 IC50 = 2.4 nM T64830 C9FED2 118963840 IC50 = 66 nM T64830 CS12JW 122179457 IC50 = 10000 nM T64830 CNGQ19 122179477 IC50 = 1530 nM T64830 C9B4DJ 122181226 Ki = 7700 nM T64830 CH1P7L 122181227 Ki = 2000 nM T64830 CV4FK8 132576638 IC50 = 3200 nM T64830 C4PNW7 132576639 IC50 = 9 nM T64830 C2VTK7 132576640 IC50 = 2800 nM T64830 C0VSA5 132576641 IC50 = 61 nM T64830 CH17SU 137631568 IC50 = 200 nM T64830 CIA6G9 137632253 IC50 > 10000 nM T64830 CQ89KJ 137638622 IC50 = 220 nM T64830 C7CI3T 137642090 IC50 = 190 nM T64830 CSKI07 137645727 IC50 = 550 nM T64830 C0N8ZV 137649134 IC50 = 150 nM T64830 C1Y7KZ 137653235 IC50 = 140 nM T64830 C82PYN 137653284 IC50 = 46 nM T64830 CLS71K 137654598 IC50 = 1000 nM T64830 CJT7B0 137658214 IC50 > 10000 nM T64830 CUV80J 137660796 IC50 = 95 nM T64830 CE79SV 138377584 IC50 = 1.1 nM T64830 COBE14 145979224 IC50 = 13 nM T64830 CE3I0L 145980226 IC50 = 28 nM T64830 CUX3P2 145980628 IC50 = 276 nM T64830 CY3L1Q 145981179 IC50 = 1 nM T64830 CY8IF4 145981627 IC50 = 0.8 nM T64830 C47WRK 145981765 IC50 = 21 nM T64830 CD6IQ0 145982284 IC50 = 8.6 nM T64830 CAE5F4 145982363 IC50 = 4.9 nM T64830 CWYP01 145989394 IC50 = 1.6 nM T64830 C7IQR6 145989603 IC50 = 78 nM T64830 CG9KC4 145989896 IC50 = 7.6 nM T64830 C3HA2T 145990504 IC50 = 19 nM T64830 CU0K2Y 145990810 IC50 = 24 nM T64830 C7H0GR 145991247 IC50 = 161 nM T64830 CYV43P 145993203 IC50 = 2.9 nM T64830 C3WLE4 145994083 IC50 = 17 nM T64830 CP0WF8 155510657 Ki > 100000 nM T64830 CW0XC1 155526536 IC50 > 1000 nM T64830 CD73TA 155526663 IC50 > 100000 nM T64830 CGXE80 155528330 Ki = 12000 nM T64830 C9QIB6 155529288 Ki = 10000 nM T64830 C9XB6L 155539840 Ki > 100000 nM T64830 C5RI8K 155541897 Ki = 4100 nM T64830 CIA72K 155543246 IC50 > 100000 nM T64830 CVR3U2 155546680 Ki = 1300 nM T64830 CGZY28 155549889 Ki = 23000 nM T64830 CLJU08 155550820 Ki = 3400 nM T64830 C89BNQ 155553012 Ki = 3900 nM T64830 C5RL2K 155565048 Ki = 5100 nM T64830 CE76TG 42637005 IC50 > 1000 nM T64830 C6ELN4 42637006 IC50 > 1000 nM T64830 CS73LG 42637433 IC50 > 1000 nM T64830 C6C3YF 45270549 IC50 > 1000 nM T64830 C9Y3BS 45270550 IC50 > 1000 nM T64830 CQC51Z 45270552 IC50 > 1000 nM T64830 CXE30U 45271377 IC50 > 1000 nM T64830 D01BWV 9802572 Ki = 2200 nM T64830 D01NID 44388055 IC50 > 1000 nM T64830 D02CQW 11847438 IC50 = 158 nM T64830 D02IXC 44403231 IC50 = 5.6 nM T64830 D02NJV 44388048 IC50 > 1000 nM T64830 D02OJQ 44388115 IC50 = 4.8 nM T64830 D02WOX 44388129 IC50 > 1000 nM T64830 D03DRL 44388045 IC50 > 1000 nM T64830 D03SXC 44388041 IC50 > 1000 nM T64830 D03VHX 44388111 IC50 > 1000 nM T64830 D04EWA 44388034 IC50 > 1000 nM T64830 D04FPW 44388024 IC50 > 1000 nM T64830 D04ORV 44388047 IC50 = 13 nM T64830 D04QBM 5311374 IC50 > 10000 nM T64830 D05COQ 11847588 IC50 = 2.7 nM T64830 D05PKR 5311375 IC50 = 0.4 nM T64830 D05XZA 44388071 IC50 > 1000 nM T64830 D06JWT 44388073 IC50 > 1000 nM T64830 D07DUF 44388130 IC50 > 1000 nM T64830 D07OSF 44388044 IC50 > 1000 nM T64830 D07WRP 15965425 Ki = 163 nM T64830 D09DAC 44388046 IC50 = 31 nM T64830 D09LHN 44311674 IC50 > 1000 nM T64830 D0A0DO 44388056 IC50 > 1000 nM T64830 D0A1XX 44388113 IC50 > 1000 nM T64830 D0BE3D 44388092 IC50 > 1000 nM T64830 D0C5RH 44388125 IC50 = 9.5 nM T64830 D0CC1P 44388042 IC50 > 1000 nM T64830 D0H0DC 44388051 IC50 > 1000 nM T64830 D0H4WH 44388128 IC50 = 5 nM T64830 D0H6LR 71717867 IC50 = 67 nM T64830 D0I9ME 44388074 IC50 > 1000 nM T64830 D0J5OY 44388022 IC50 = 8.6 nM T64830 D0M5LA 44388050 IC50 > 1000 nM T64830 D0N2MA 44388103 IC50 > 1000 nM T64830 D0N4LH 44388065 IC50 > 1000 nM T64830 D0O4GU 44403230 Ki = 13.1 nM T64830 D0P6ZZ 10581102 IC50 > 1000 nM T64830 D0R0OX 44388102 IC50 > 1000 nM T64830 D0R4IS 44388131 IC50 > 1000 nM T64830 D0S7YR 44388059 IC50 > 1000 nM T64830 D0T5RO 16129706 EC50 = 0.065 nM T64830 D0W0AF 44388072 IC50 > 1000 nM T64830 D0WG0O 44388049 IC50 > 1000 nM T64830 D0Z0OF 44388094 IC50 > 1000 nM T64830 D0Z1XY 44388064 IC50 > 1000 nM T64830 D0Z3LZ 44388023 IC50 = 43 nM T20953 D03HUX 49792852 IC50 > 10000 nM T20953 CU3RF1 45139989 IC50 > 10000 nM T20953 CQGZ06 45139991 IC50 > 10000 nM T20953 C7ON5A 46233287 IC50 > 10000 nM T20953 CF91RS 49843531 IC50 > 10000 nM T20953 C2Y6QS 50938552 IC50 > 10000 nM T20953 C9NYP4 51036677 IC50 > 10000 nM T20953 C4WRY3 51037112 IC50 > 10000 nM T20953 CRI28Z 51037948 IC50 > 10000 nM T20953 CCN01X 71547862 IC50 > 10000 nM T20953 CYB9A4 72202967 IC50 = 2000 nM T20953 CY0UC4 90645194 IC50 > 10000 nM T20953 C16TDG 90655893 IC50 = 500 nM T20953 CY7BI2 118706214 IC50 > 10000 nM T20953 D09BXA 72202254 IC50 = 5 nM T20953 D0F9DD 72203102 IC50 = 30 nM T20953 D0JP7S 72202696 IC50 = 9 nM T20953 D0P4YY 72202697 IC50 = 6 nM T21038 CORM50 584781 IC50 > 20000 nM T21038 C2VZH3 647508 IC50 = 940 nM T21038 C43VDF 743900 IC50 = 7700 nM T21038 C3VK0C 746711 IC50 = 6300 nM T21038 CF92JY 755364 IC50 > 20000 nM T21038 C27RMY 814607 IC50 = 1220 nM T21038 CYOS57 909915 IC50 = 790 nM T21038 CQ04VL 1088429 IC50 > 20000 nM T21038 C83ECX 1088431 IC50 = 18000 nM T21038 C0BJ4Y 1088435 IC50 = 2800 nM T21038 CBP2S9 1088438 IC50 = 560 nM T21038 CSY32B 1088439 IC50 = 90 nM T21038 CP40AO 1106348 IC50 = 3440 nM T21038 CWG9X3 1106353 IC50 = 830 nM T21038 C31QOG 1106356 IC50 = 1030 nM T21038 CPM4V8 1106360 IC50 = 1130 nM T21038 CRN6H2 1106361 IC50 = 150 nM T21038 CKLU94 1142837 IC50 = 3110 nM T21038 C5JTM8 1360138 IC50 = 510 nM T21038 CYO14C 3025920 IC50 = 2200 nM T21038 CJ72HY 3025945 IC50 = 14000 nM T21038 C9UOZ1 4782333 IC50 = 3300 nM T21038 CETX38 5310346 IC50 = 1540 nM T21038 C0ZI8N 14783456 IC50 = 5740 nM T21038 CW6RP7 15992998 IC50 = 17400 nM T21038 C5C2LS 15994862 IC50 > 20000 nM T21038 C1DEF3 15996790 IC50 = 2570 nM T21038 C8Y9WJ 16000292 IC50 > 20000 nM T21038 CNIO43 16002787 IC50 = 1870 nM T21038 C4ZPG6 16021204 IC50 = 3630 nM T21038 C5PUD1 19062910 IC50 > 20000 nM T21038 C1ZAB6 20853147 IC50 = 11150 nM T21038 CR0EV3 20853151 IC50 = 4420 nM T21038 C65QXZ 20853209 IC50 > 20000 nM T21038 CGW08K 20901603 IC50 = 5600 nM T21038 C5VKZ1 20901630 IC50 > 20000 nM T21038 CGJ05B 20901660 IC50 = 10260 nM T21038 CG9Y7Z 20901691 IC50 = 510 nM T21038 C0CGA3 26528163 IC50 > 20000 nM T21038 CYV4Q6 41455001 IC50 > 20000 nM T21038 CX9B7O 41455005 IC50 > 20000 nM T21038 C9EC6T 42370913 IC50 > 20000 nM T21038 CH49XR 44182107 IC50 > 20000 nM T21038 CJ6G9A 44182108 IC50 > 20000 nM T21038 CEY1Z0 44182132 IC50 = 1700 nM T21038 CNS3C2 44182143 IC50 = 1010 nM T21038 C2OMP6 44182144 IC50 = 2000 nM T21038 CA9GE5 44182145 IC50 = 260 nM T21038 C65SAT 44182146 IC50 = 5760 nM T21038 C8R2GZ 44182147 IC50 > 20000 nM T21038 CY02GM 44182148 IC50 > 20000 nM T21038 CU1X7V 44182149 IC50 = 240 nM T21038 CQL3Y2 44182150 IC50 > 20000 nM T21038 C6AUS5 44229052 IC50 > 20000 nM T21038 CG6YQ2 44229053 IC50 = 1610 nM T21038 CH6QI1 44229054 IC50 > 20000 nM T21038 CJWQ24 44229055 IC50 = 80 nM T21038 C7QTA4 44229056 IC50 > 20000 nM T21038 CEA0F8 44229057 IC50 = 10600 nM T21038 CVX8C7 44229058 IC50 > 20000 nM T21038 CU98HG 44229059 IC50 > 20000 nM T21038 CZ2X0O 44229060 IC50 > 20000 nM T21038 CT28PV 44229066 IC50 = 2700 nM T21038 C3PXS0 44229067 IC50 > 20000 nM T21038 COAV34 44236880 IC50 > 20000 nM T21038 CDNB26 44251466 IC50 > 20000 nM T21038 CX84MR 44251468 IC50 = 6500 nM T21038 CA9CN4 44251469 IC50 > 20000 nM T21038 C9XJI7 44251470 IC50 = 5870 nM T21038 CAD8P0 44251474 IC50 > 20000 nM T21038 CA5JC4 44251475 IC50 > 20000 nM T21038 CNP1T4 44412097 IC50 = 19800 nM T21038 CC1AV6 44543518 IC50 > 20000 nM T21038 CAZE43 51349461 EC50 > 100 nM T21038 CD4LS9 51349463 EC50 > 100 nM T21038 CTJP03 51349605 EC50 = 1.73 nM T21038 C2KNG7 51349607 EC50 > 100 nM T21038 C4KV3P 51349609 EC50 = 0.37 nM T21038 CCL12D 51349747 EC50 = 0.57 nM T21038 CZ56SP 51349749 EC50 = 0.96 nM T21038 CUB5O9 51349877 EC50 = 0.2 nM T21038 CDK4Q6 51349879 EC50 = 0.0015 nM T21038 CR8KN3 51349881 EC50 = 0.12 nM T21038 CBQU21 51349883 EC50 = 0.622 nM T21038 CV39UM 51350010 EC50 = 0.027 nM T21038 C0S2IT 51350012 EC50 = 0.066 nM T21038 C6E8YZ 51350014 EC50 = 0.826 nM T21038 C05EZQ 51350016 EC50 = 0.134 nM T21038 C9QW1R 51350018 EC50 = 0.238 nM T21038 CT12PX 51350155 EC50 = 0.55 nM T21038 C9BLD4 51350157 EC50 = 0.58 nM T21038 CG62FV 51350159 EC50 = 0.069 nM T21038 CZM37E 51350161 EC50 = 0.181 nM T21038 CIA85X 51350163 EC50 = 0.145 nM T21038 CDGR40 51350165 EC50 = 0.504 nM T21038 CN6AV9 51350167 EC50 = 0.39 nM T21038 CC8OV3 51350287 EC50 = 0.023 nM T21038 C1ELK2 70683344 IC50 > 20000 nM T21038 CPD08T 70693845 IC50 = 16300 nM T21038 C2Y3WL 102369397 IC50 = 400 nM T21038 CS79JV 117889777 IC50 > 10000 nM T21038 CCL2R0 117907988 IC50 > 10000 nM T21038 C46GHP 117908214 IC50 > 10000 nM T21038 C7SK6U 117908215 IC50 > 10000 nM T21038 C6WXO0 118709778 IC50 = 800 nM T21038 CRM0Q5 118709779 IC50 = 1600 nM T21038 CDL14S 118709780 IC50 = 1300 nM T21038 CKD73Y 118709781 IC50 = 3400 nM T21038 C0ZO1K 118709782 IC50 = 200 nM T21038 CBF7C8 118711983 IC50 > 10000 nM T21038 C2TE9N 118711985 IC50 > 10000 nM T21038 C1LDN8 137631490 IC50 = 580 nM T21038 CE73UJ 137631857 IC50 = 1370 nM T21038 C5DIX0 137632307 IC50 = 580 nM T21038 CX1T9D 137632432 IC50 = 1610 nM T21038 CN43SO 137632600 IC50 = 2900 nM T21038 CZ29XV 137633122 IC50 = 2360 nM T21038 C3LXK0 137635005 IC50 = 2810 nM T21038 C7WC0M 137635525 IC50 = 1300 nM T21038 CB7JM9 137636367 IC50 = 2370 nM T21038 C2D8EO 137636592 IC50 = 1330 nM T21038 CS9P3G 137637882 IC50 = 1290 nM T21038 C1ZCB7 137638553 IC50 = 3990 nM T21038 CRY36U 137639197 IC50 = 1290 nM T21038 CE5WD2 137639318 IC50 = 8620 nM T21038 CU31EO 137640364 IC50 = 1390 nM T21038 CXO01A 137642351 IC50 = 1060 nM T21038 CH85VU 137643081 IC50 = 1270 nM T21038 C1H9WD 137644120 IC50 = 940 nM T21038 C3NDC2 137645474 IC50 = 1930 nM T21038 C0D9ZT 137645928 IC50 = 1110 nM T21038 CZ92HB 137646848 IC50 = 2360 nM T21038 C3ZWY0 137650229 IC50 = 430 nM T21038 CH78YX 137652947 IC50 = 1110 nM T21038 COU32W 137653192 IC50 = 1550 nM T21038 CJQT49 137653516 IC50 = 1960 nM T21038 CHC9X4 137655226 IC50 = 1330 nM T21038 C31EUD 137656156 IC50 = 4950 nM T21038 CY0V9Z 137656864 IC50 = 1160 nM T21038 C3ZS8Y 137657750 IC50 = 610 nM T21038 CT28EF 137660858 IC50 = 580 nM T21038 C5WJ0C 155521741 IC50 = 15700 nM T21038 CGN5P7 155529528 IC50 = 15000 nM T21038 CZ0NQ1 155536959 IC50 = 7780 nM T21038 CQT7U2 155546687 IC50 = 16000 nM T21038 CY72AR 155566972 IC50 = 9220 nM T99347 D00ENY 33032 Ki = 390 nM T99347 D0X9RY 243 EC50 > 10000 nM T99347 D04QKU 11438771 IC50 = 7 nM T99347 D0G5PF 9926832 Ki = 5.6 nM T99347 D0I5TL 44557636 IC50 = 20 nM T99347 D06LYZ 11559235 IC50 = 342 nM T99347 D0AK4X 74222037 IC50 = 50 nM T99347 D0CI3E 50990953 Ki = 6.8 nM T99347 D0D3GL 137662068 IC50 = 75 nM T99347 D0D4OW 57338826 EC50 > 25000 nM T99347 D0FS2X 90646678 Ki = 3.981 nM T99347 D0KG5I 118204326 IC50 = 28.7 nM T99347 D0LU9X 74221950 IC50 = 38 nM T99347 D0PJ8X 71562840 IC50 = 410 nM T99347 D0RU0W 137639643 IC50 = 32 nM T99347 D0XX9N 137637236 IC50 = 46 nM T99347 D04JQR 5311261 IC50 > 300000 nM T99347 D09XHI 9879103 IC50 = 13.4 nM T99347 D0E3SD 9838729 IC50 = 7.6 nM T99347 D0U5CS 213056 EC50 > 100000 nM T99347 D0ZV0R 16660135 IC50 = 7000 nM T99347 C0MLE4 1217 Ki = 14000 nM T99347 CL8RX5 1222 Ki > 2000000 nM T99347 COC91V 10255 EC50 = 33600 nM T99347 CCD82P 64809 EC50 > 10000 nM T99347 C9H6OS 92136 Ki > 1000000 nM T99347 CUT07K 177491 Ki = 54000 nM T99347 CNQ5I7 342595 EC50 = 75 nM T99347 CWBV63 342596 EC50 = 20 nM T99347 CO9KU6 443586 Ki = 1900 nM T99347 C6CA0S 623968 EC50 = 970 nM T99347 CI96OA 650707 IC50 = 116 nM T99347 CPA10R 657896 IC50 > 100000 nM T99347 C4HP6J 661617 IC50 > 10000 nM T99347 CEI29J 665694 IC50 > 100000 nM T99347 C9DX2A 685051 IC50 = 2570 nM T99347 CGQ2R3 692972 IC50 = 9600 nM T99347 C18QMW 695758 IC50 > 10000 nM T99347 C9P2IQ 699222 IC50 > 100000 nM T99347 CM3R2L 702923 IC50 = 1700 nM T99347 CT43JC 705823 IC50 = 118 nM T99347 CCBT27 720143 Ki > 10000 nM T99347 CIJ7U2 744275 IC50 = 890 nM T99347 CY8XQ1 750619 IC50 > 10000 nM T99347 C9IRB2 763879 IC50 = 436 nM T99347 C0OCI1 769041 IC50 = 1540 nM T99347 CCX4T0 778172 Ki = 410 nM T99347 CHWG63 789864 IC50 = 540 nM T99347 CK81OA 812404 IC50 = 600 nM T99347 CNU37V 812406 IC50 = 300 nM T99347 CWG31F 812407 IC50 = 500 nM T99347 CVSO71 812500 IC50 = 200 nM T99347 C6I9LM 812501 IC50 = 3100 nM T99347 C69PWH 812702 IC50 = 1800 nM T99347 C2LPI1 812703 IC50 > 10000 nM T99347 CB0S6U 812719 IC50 = 300 nM T99347 CDIV53 812720 IC50 = 80 nM T99347 C0FM6O 867096 IC50 = 236 nM T99347 C2Z6CA 921213 IC50 = 30000 nM T99347 C8WB4L 944643 IC50 = 492 nM T99347 CK98RL 1069776 IC50 = 1810 nM T99347 CUA1T7 1142605 IC50 = 1.1 nM T99347 C7VCI2 1208332 IC50 > 3000 nM T99347 CKT3N7 1284324 IC50 > 100000 nM T99347 C0UT9W 1336785 EC50 = 720 nM T99347 CJC8S2 1364364 EC50 = 776.25 nM T99347 C9GJS3 1431783 IC50 > 10000 nM T99347 CAU1W0 1441195 IC50 = 10000 nM T99347 C5MDN9 1441201 IC50 = 310 nM T99347 C1MTA0 1441202 IC50 = 5400 nM T99347 CXO3M6 1441208 IC50 = 1800 nM T99347 CF3QH0 1447824 IC50 = 2300 nM T99347 C9BG2F 1447967 IC50 > 10000 nM T99347 C8BKA4 1486708 IC50 = 142 nM T99347 C7X8KU 1489964 IC50 > 10000 nM T99347 CNI89V 1617110 Ki > 1000000 nM T99347 CUP21W 2725933 IC50 = 1250 nM T99347 C5F8YH 2733519 EC50 = 105000 nM T99347 CLU24Y 2818849 EC50 = 2500 nM T99347 CM5TO1 2837010 Ki = 7000 nM T99347 CH58DV 2839591 IC50 > 10000 nM T99347 CC3D9F 2861965 IC50 = 990 nM T99347 CB4QY6 2955988 IC50 > 30000 nM T99347 CWT86X 3011435 IC50 = 105 nM T99347 CDM78G 3156022 IC50 = 443 nM T99347 CRN67W 3354176 Ki > 10000 nM T99347 CLFH17 3655510 IC50 > 31622.78 nM T99347 CJZC03 3773077 IC50 = 598 nM T99347 C57BKY 3796302 IC50 = 2300 nM T99347 CP5C1A 3931705 Ki > 100000 nM T99347 CLNV31 4107180 IC50 > 10000 nM T99347 CJK71C 4287026 EC50 = 3100 nM T99347 CXN2P8 4384110 EC50 = 1380 nM T99347 COJV81 4521898 EC50 = 165.96 nM T99347 CZ1Q5P 4694355 Ki > 1000000 nM T99347 CY1NB7 5075788 IC50 = 63 nM T99347 CRS7U5 5075956 IC50 = 373 nM T99347 C05WNA 5310956 Ki = 3100 nM T99347 CGMN04 5311262 Ki = 470 nM T99347 CB8Z2W 5640190 Ki = 306.8 nM T99347 C2T5NV 5640191 Ki = 310.2 nM T99347 C3QR9Z 5640192 Ki = 108.2 nM T99347 C1M7AH 5640487 Ki = 201.2 nM T99347 C87WCF 6457595 EC50 = 350 nM T99347 CEA9F2 6463470 IC50 = 845 nM T99347 CZ3G8M 6603702 IC50 > 1000000 nM T99347 C7J6KQ 6604704 EC50 > 300000 nM T99347 CD68LI 6604795 Ki > 1000000 nM T99347 C80RDG 7184909 Ki = 198 nM T99347 CYZ57U 7298720 IC50 = 2500 nM T99347 C5OLQ0 9554216 IC50 = 620 nM T99347 CL7Y9V 9570595 IC50 > 10000 nM T99347 CIA9B5 9794218 IC50 = 5 nM T99347 C5WAT4 9815955 Ki > 100000 nM T99347 CL8JI1 9837114 EC50 > 1000000 nM T99347 CEF2X1 9837457 IC50 = 31.62 nM T99347 C8NWE5 9844204 Ki = 3400 nM T99347 CPQ47V 9858082 IC50 = 2859 nM T99347 C0D3WM 9878140 IC50 > 10000 nM T99347 CW8JL3 9881610 IC50 = 154 nM T99347 CDEN35 9902170 IC50 = 124 nM T99347 C0CB7T 9921211 IC50 = 690 nM T99347 CURS80 9926060 IC50 = 274 nM T99347 CD9MQ4 9944756 IC50 = 737 nM T99347 C8XNY7 9945473 IC50 = 17 nM T99347 C69CEB 9948499 IC50 = 700 nM T99347 CT7BR0 9965311 Ki = 69 nM T99347 C0GN6F 10012356 Ki = 490000 nM T99347 C7EJ5D 10013513 EC50 = 11000 nM T99347 CUN9V7 10036599 IC50 > 300000 nM T99347 CLY69G 10039170 IC50 = 2 nM T99347 CGLR38 10059467 EC50 = 398.11 nM T99347 C0OI6Q 10063269 IC50 = 70 nM T99347 CG4P8U 10063270 IC50 = 28 nM T99347 C2BG6C 10085660 Ki = 22 nM T99347 CW8U5B 10125821 IC50 = 309 nM T99347 CONB04 10130339 IC50 = 10 nM T99347 C41XGZ 10150237 IC50 = 451 nM T99347 COCK70 10150315 IC50 = 229 nM T99347 CWV78P 10192780 IC50 = 6150 nM T99347 C1WR6I 10192781 IC50 = 210 nM T99347 CLE19O 10193697 IC50 = 16 nM T99347 C9XQK6 10198133 EC50 > 100000 nM T99347 CL4NP9 10198359 EC50 = 1000 nM T99347 CCB29V 10198810 IC50 = 100 nM T99347 CSX82D 10236196 IC50 = 980 nM T99347 CFDX64 10241509 EC50 > 300000 nM T99347 CZ7A5Y 10263168 Ki = 97000 nM T99347 C6M8JC 10266278 IC50 = 12 nM T99347 CAX8R2 10269322 IC50 = 13 nM T99347 CDWT20 10285979 IC50 > 10000 nM T99347 CA7PI3 10285980 IC50 = 80 nM T99347 CWP90L 10286300 IC50 = 63 nM T99347 CC8K7G 10291336 IC50 = 22 nM T99347 CBY57U 10308407 IC50 = 334 nM T99347 C0ZT5K 10308416 IC50 = 2102 nM T99347 C8W2LA 10308678 IC50 = 461 nM T99347 CX12HM 10330132 Ki > 1000000 nM T99347 CWZ27Y 10331863 IC50 = 17 nM T99347 CZ09YG 10358265 IC50 > 300000 nM T99347 CQ1L0O 10359073 Ki > 300000 nM T99347 CXFL79 10382361 Ki = 0.5 nM T99347 CYL91R 10456810 IC50 > 100000 nM T99347 C3KHU7 10465017 EC50 > 1000000 nM T99347 CK9MN4 10465478 EC50 = 190000 nM T99347 C9ET6D 10470570 Ki = 32 nM T99347 CH9VN3 10560963 EC50 = 91000 nM T99347 CQTF38 10775369 EC50 = 57000 nM T99347 C9BK1A 10846649 EC50 = 720 nM T99347 C2HT9A 11149253 IC50 = 556 nM T99347 CJ5A6T 11150516 IC50 = 134 nM T99347 C0ZUT6 11152155 EC50 = 200 nM T99347 CQ7S8F 11164167 EC50 = 30 nM T99347 CIX7Z1 11171896 IC50 = 165 nM T99347 CFM4Q1 11172830 IC50 = 46 nM T99347 CFE92I 11175693 EC50 > 10000 nM T99347 CSNA95 11183505 IC50 = 3536 nM T99347 CV3C9Z 11185714 IC50 = 862 nM T99347 C0PLH7 11188537 EC50 = 2100 nM T99347 C21FTG 11195510 IC50 = 32 nM T99347 C0EG2L 11196589 IC50 = 43 nM T99347 CU5Q9Z 11200691 EC50 = 330 nM T99347 C0WRB3 11207899 IC50 = 416 nM T99347 C3APV5 11218324 IC50 = 223 nM T99347 CH78IP 11219258 IC50 = 5 nM T99347 C8H1ZI 11220495 IC50 = 193 nM T99347 CTB6X3 11220891 IC50 = 11 nM T99347 CVFG01 11221928 EC50 > 10000 nM T99347 CDY95C 11222596 EC50 = 10 nM T99347 COM6P1 11231404 IC50 = 1900 nM T99347 CKT3V0 11232032 IC50 = 12 nM T99347 C0GSF6 11233624 EC50 = 13900 nM T99347 C5TFV7 11234162 EC50 = 40 nM T99347 CN38LI 11234371 EC50 = 2300 nM T99347 C0REF5 11241984 IC50 = 7 nM T99347 C18VSQ 11246786 EC50 = 19 nM T99347 CFQ20E 11253176 IC50 = 3000 nM T99347 C06TSN 11256060 IC50 = 210 nM T99347 CG8HC7 11256656 IC50 = 80 nM T99347 C04MKF 11265885 IC50 = 36 nM T99347 C6XD1J 11265888 IC50 = 158 nM T99347 C1MKP9 11267265 IC50 = 126 nM T99347 CDC6I1 11279648 EC50 = 90 nM T99347 CL5X1Y 11290518 IC50 = 103 nM T99347 CL9MT5 11299520 IC50 = 119 nM T99347 C24NHT 11311245 IC50 = 11 nM T99347 CW67DI 11323067 IC50 = 83 nM T99347 CUV4Z0 11325594 IC50 = 2300 nM T99347 CD23KN 11333966 IC50 = 22 nM T99347 CDI71C 11334544 IC50 = 145 nM T99347 C80BLF 11336477 IC50 = 37 nM T99347 CTWH72 11345889 IC50 = 174 nM T99347 CAC7N1 11345906 IC50 = 102 nM T99347 CKBE95 11346332 IC50 = 6200 nM T99347 CR6UH2 11347767 IC50 = 45 nM T99347 CS8NY9 11351706 EC50 = 470000 nM T99347 C7C1QS 11356950 IC50 = 2700 nM T99347 C3MD9R 11357227 IC50 = 455 nM T99347 C2KFP6 11358285 IC50 = 15 nM T99347 CGH3Y5 11368190 IC50 = 40 nM T99347 CA0N8R 11368523 IC50 = 1600 nM T99347 C1BAS3 11369816 IC50 = 870 nM T99347 C0NKF1 11370077 IC50 = 1520 nM T99347 CGVO76 11370949 IC50 = 80 nM T99347 C5W3AY 11371383 EC50 = 1800 nM T99347 CR5D9O 11379364 IC50 = 6728 nM T99347 CW86BH 11381681 IC50 = 18 nM T99347 C0JH9E 11382254 EC50 = 200 nM T99347 C25GLF 11382452 IC50 = 390 nM T99347 CIS36X 11396858 EC50 = 930 nM T99347 CIZ8U9 11402081 IC50 = 254 nM T99347 C4DTO3 11402257 IC50 = 8 nM T99347 C4CUW5 11402852 IC50 = 22 nM T99347 C2OIW4 11405070 EC50 = 290 nM T99347 C4HR0W 11413259 IC50 = 458 nM T99347 CC51BG 11414108 IC50 = 397 nM T99347 C8IH7J 11414998 IC50 = 118 nM T99347 C6WIO7 11415160 IC50 = 12 nM T99347 CRME92 11415580 IC50 = 47 nM T99347 C8XDS1 11418750 EC50 = 1500 nM T99347 CX2JK6 11448439 IC50 = 17 nM T99347 CQR52H 11450419 IC50 = 550 nM T99347 C6WJR7 11451163 EC50 = 20 nM T99347 CSU48Y 11452267 EC50 = 1500 nM T99347 CLJK95 11458873 IC50 = 497 nM T99347 CHP0B6 11460538 IC50 = 21 nM T99347 CCW5A2 11462332 EC50 = 30 nM T99347 CW7JA2 11463475 EC50 = 245 nM T99347 CX7Q2S 11473141 IC50 = 28 nM T99347 C9K8XT 11481862 Ki = 1.7 nM T99347 C5K8AH 11492398 IC50 > 10000 nM T99347 CT9LY1 11492417 IC50 > 10000 nM T99347 CY1GT7 11492602 IC50 > 10000 nM T99347 C90BXG 11493585 IC50 = 901 nM T99347 CWQU24 11493897 IC50 = 592 nM T99347 C79QDF 11499598 IC50 = 228 nM T99347 CR5KB3 11500296 IC50 = 10.2 nM T99347 CTB4K0 11501188 IC50 > 100000 nM T99347 CI6G2R 11501465 IC50 = 344 nM T99347 C7C1UQ 11508375 Ki = 67 nM T99347 CD4H3R 11508696 IC50 > 10000 nM T99347 CB1S3Q 11514058 IC50 > 10000 nM T99347 CS27NI 11514100 IC50 = 19.2 nM T99347 CTA5R7 11514153 IC50 = 426 nM T99347 CD97RY 11515445 Ki = 31 nM T99347 C60PZU 11515679 IC50 > 100000 nM T99347 CY8SI0 11515957 IC50 = 179 nM T99347 CJ3HW2 11521435 IC50 = 192 nM T99347 CJE20A 11522172 IC50 = 2340 nM T99347 CLA0Q4 11529197 IC50 > 10000 nM T99347 CQNE82 11530673 IC50 = 2040 nM T99347 CY90XO 11530971 IC50 = 4530 nM T99347 CBNZ75 11537426 IC50 = 488 nM T99347 C9FGB7 11537767 IC50 > 100000 nM T99347 C5TG6U 11537814 IC50 > 100000 nM T99347 CL84DM 11543451 IC50 > 10000 nM T99347 CSFO10 11552320 IC50 = 3540 nM T99347 CT9RC0 11558879 Ki = 9 nM T99347 CZVQ09 11560185 IC50 > 100000 nM T99347 C8OTP6 11564911 IC50 > 10000 nM T99347 CV7FE9 11565466 IC50 > 100000 nM T99347 CWS27I 11565576 IC50 > 10000 nM T99347 CE2P8Y 11566478 IC50 = 2160 nM T99347 C6XH5Z 11574901 IC50 = 1250 nM T99347 CXIU67 11579421 IC50 = 1093 nM T99347 C23SQX 11581985 IC50 > 100000 nM T99347 CTBF56 11582178 IC50 > 100000 nM T99347 CN91LK 11586574 IC50 = 833 nM T99347 CW8M5V 11588590 IC50 = 4620 nM T99347 CAU3J7 11594013 IC50 > 10000 nM T99347 C5Z9KA 11594849 IC50 > 100000 nM T99347 CUOP90 11595030 Ki = 81 nM T99347 CGX8F6 11596869 EC50 > 12500 nM T99347 CT64YE 11608542 IC50 = 68.6 nM T99347 C3J6UO 11609353 IC50 = 1160 nM T99347 C3VI5L 11616166 IC50 = 266 nM T99347 C1ZX5N 11618305 IC50 = 2.2 nM T99347 CVL43G 11623479 IC50 = 162 nM T99347 CMBS38 11631279 IC50 > 100000 nM T99347 CP6WU2 11637242 IC50 = 45.5 nM T99347 C8CKV1 11638418 Ki = 44 nM T99347 C9F3WR 11639176 IC50 = 2570 nM T99347 CCET62 11639210 IC50 > 100000 nM T99347 CD5Q9A 11652895 IC50 > 100000 nM T99347 CVYR03 11654379 IC50 = 901 nM T99347 CU58GV 11660511 IC50 = 2100 nM T99347 C1P3XR 11660540 IC50 > 100000 nM T99347 C0MOJ5 11661106 IC50 > 100000 nM T99347 C3RBF5 11665983 IC50 > 10000 nM T99347 CJ85FI 11666576 IC50 > 100000 nM T99347 C2B3CR 11667061 Ki = 13 nM T99347 CGR90L 11667270 IC50 = 11300 nM T99347 CRG5I8 11673933 IC50 = 225 nM T99347 CO3X5A 11674352 IC50 = 3900 nM T99347 CSJ53G 11680198 IC50 = 2950 nM T99347 C6ZB8C 11681575 IC50 = 5960 nM T99347 C0VRM1 11681680 IC50 = 2160 nM T99347 C65FWA 11681681 IC50 > 100000 nM T99347 CTAP95 11682046 IC50 > 100000 nM T99347 CLVO83 11682866 IC50 > 100000 nM T99347 C2C4WA 11687246 IC50 > 10000 nM T99347 CD1O9I 11688761 IC50 = 16 nM T99347 CJCZ59 11688880 IC50 > 100000 nM T99347 C3Z4MV 11694640 IC50 = 413 nM T99347 C97SMI 11695588 IC50 = 650 nM T99347 C1ILY6 11695769 IC50 > 100000 nM T99347 CF6LG4 11695894 IC50 = 40 nM T99347 CR5B3L 11696595 IC50 = 154 nM T99347 CND69H 11702918 IC50 = 816 nM T99347 C5HFM9 11703031 IC50 > 100000 nM T99347 CX7SQ9 11708662 IC50 = 2020 nM T99347 C95EAP 11709446 IC50 > 10000 nM T99347 C2KF0Y 11709877 Ki = 111 nM T99347 CS0A4X 11717278 IC50 > 100000 nM T99347 CY2VL6 11717319 IC50 > 100000 nM T99347 C42RJY 11735574 IC50 = 81 nM T99347 C0IXK9 11737347 IC50 = 281 nM T99347 C7CM4E 11750147 EC50 = 260 nM T99347 CASI54 11768848 EC50 > 1000000 nM T99347 CX7VJ1 11769227 IC50 = 97 nM T99347 C47WVT 11769507 IC50 = 13 nM T99347 C9TUB7 11771968 IC50 = 90 nM T99347 CP7QF3 11772069 IC50 = 1100 nM T99347 C96YUT 11820180 Ki = 36000 nM T99347 CJ4WL9 15207262 IC50 > 100000 nM T99347 CSW38G 15420544 EC50 = 346.74 nM T99347 C41MVD 15942645 IC50 = 10 nM T99347 CR8J1L 15942646 IC50 = 20 nM T99347 C8PWY3 15949470 Ki = 1 nM T99347 CPC09T 15985249 IC50 = 2800 nM T99347 CETV92 16065021 IC50 = 20 nM T99347 CJEN28 16117979 IC50 > 10000 nM T99347 C64FAY 16118120 IC50 = 1201 nM T99347 CSLK82 16118121 IC50 = 1321 nM T99347 C3WI2G 16118122 IC50 = 515 nM T99347 C6X3ED 16118123 IC50 = 7844 nM T99347 C4R1BK 16118124 IC50 > 10000 nM T99347 C4X6EZ 16118680 IC50 > 100000 nM T99347 CE0VB6 16118681 IC50 > 1000 nM T99347 CY4I3R 16118682 IC50 > 1000 nM T99347 CZ1Y2D 16118812 IC50 > 1000 nM T99347 C87ZLF 16118813 IC50 > 1000 nM T99347 C1T7IZ 16124095 Ki = 204.17 nM T99347 C45BPW 16202228 Ki = 52 nM T99347 CASK57 16584098 IC50 = 93.6 nM T99347 C0M8NP 16659645 IC50 > 1000 nM T99347 C7RHT2 16659646 IC50 > 10000 nM T99347 C8ZXU6 16659804 IC50 > 1000 nM T99347 C71WGT 16659805 IC50 > 1000 nM T99347 CWT36L 16659966 IC50 = 702 nM T99347 C8IX9D 16659968 IC50 = 609 nM T99347 C80LVT 16660140 IC50 = 9200 nM T99347 CZ2IS9 16660294 IC50 = 7900 nM T99347 CI86GL 16660467 IC50 > 10000 nM T99347 CSX4P9 16662881 IC50 = 3 nM T99347 C5L0MD 16664610 IC50 = 60 nM T99347 CFK3Y4 16730836 IC50 = 160 nM T99347 CJ2X4N 16735660 IC50 = 132 nM T99347 C6NZ2I 16736016 IC50 = 85 nM T99347 CJA3N2 16736017 IC50 = 52 nM T99347 C6XQ2O 16736020 IC50 = 80 nM T99347 C4VBJ7 16736021 IC50 = 1890 nM T99347 C5EJ6G 16736023 IC50 = 8900 nM T99347 CJ0HQ4 16736032 IC50 = 96 nM T99347 CORG05 16736033 IC50 = 312 nM T99347 C5Y8BS 16955911 EC50 = 170 nM T99347 CY37IV 16955920 EC50 = 58 nM T99347 CP69WV 16955923 EC50 = 8.8 nM T99347 CQBS15 16955925 EC50 > 10000 nM T99347 C1W9ON 16955951 IC50 = 3520 nM T99347 CGOE91 16955975 EC50 = 240 nM T99347 C5DKZ8 16956771 EC50 = 5.1 nM T99347 C6FE3O 16956776 EC50 > 10000 nM T99347 CW3GE4 16956789 EC50 = 310 nM T99347 C7PS0F 17228330 IC50 = 496 nM T99347 C04GUC 17758443 Ki = 49000 nM T99347 C0Z2XO 17758444 Ki = 67000 nM T99347 CGZF13 17758445 Ki > 300000 nM T99347 C1GSZ4 17758449 Ki = 55000 nM T99347 CZW76I 17758450 Ki > 300000 nM T99347 CT64UF 17758554 Ki = 81000 nM T99347 C3X6WB 17758555 Ki > 300000 nM T99347 C1AD2J 17758556 Ki > 300000 nM T99347 CN6IP3 17915602 IC50 = 940 nM T99347 CL3E1K 18107205 Ki = 7290 nM T99347 CS5B7A 18138918 Ki = 440 nM T99347 COI7N2 18763270 IC50 = 7 nM T99347 C6FTH4 19705292 IC50 = 820 nM T99347 C7W5BK 19851586 IC50 = 872 nM T99347 C1K5ZA 20763893 Ki = 60.7 nM T99347 CIW73R 21942491 IC50 = 23 nM T99347 CZC8U4 21942492 IC50 = 61 nM T99347 CD6PM1 22268047 EC50 = 103000 nM T99347 CQU96V 22583268 EC50 = 398.11 nM T99347 C0K9DR 22884216 IC50 = 195000 nM T99347 CLN7Z9 23133570 IC50 = 580 nM T99347 CTQ5X8 23634169 IC50 > 3000 nM T99347 CW2PD7 23634249 IC50 > 3000 nM T99347 CKL4B6 23634254 IC50 > 3000 nM T99347 C5E1DJ 23634325 IC50 > 3000 nM T99347 CX3BC2 23634326 IC50 > 3000 nM T99347 CZ4EC2 23655076 IC50 > 100000 nM T99347 CJ18UB 23657393 IC50 > 1000 nM T99347 CD1A4H 23725275 IC50 = 430 nM T99347 CFBP69 23725277 IC50 = 530 nM T99347 CK4P1X 23725388 IC50 = 10000 nM T99347 C6SJ0C 23725442 IC50 = 105 nM T99347 CR9EA6 23725445 IC50 = 87 nM T99347 C7DO2G 23725537 IC50 = 48 nM T99347 CMT69Q 23725540 IC50 = 140 nM T99347 C1Z7GN 23725592 IC50 = 420 nM T99347 CX1LK9 23725593 IC50 = 250 nM T99347 CWFI98 23725594 IC50 = 2300 nM T99347 CVZ09F 23725698 IC50 = 90 nM T99347 C3K0OP 23725701 IC50 = 390 nM T99347 CWGD32 23725754 IC50 = 1400 nM T99347 C53NCU 23725758 IC50 = 240 nM T99347 CUC23M 23725809 IC50 = 40 nM T99347 C6VHK1 23725810 IC50 = 40 nM T99347 CMS4Q5 23725812 IC50 = 16 nM T99347 C7W2LT 23725862 IC50 = 5 nM T99347 CCS5N3 23725974 IC50 = 64 nM T99347 C1JR7P 24246632 Ki = 7580 nM T99347 CJWM19 24762469 EC50 = 1280 nM T99347 CX9VZ2 24762470 EC50 = 10300 nM T99347 C0CXU2 24762868 EC50 = 1100 nM T99347 C2SW9X 24762950 EC50 = 1000 nM T99347 CU2C5L 24762951 EC50 = 7100 nM T99347 C5CN8X 24762952 EC50 = 1100 nM T99347 CWCR46 24762955 EC50 = 300 nM T99347 C0XO5U 24763199 EC50 = 180 nM T99347 C91XQC 24763201 EC50 = 270 nM T99347 C5S6PG 24763202 EC50 = 310 nM T99347 CPY95O 24763203 EC50 = 1090 nM T99347 CD8C0H 24763283 EC50 = 4600 nM T99347 CM16AG 24763370 EC50 = 1300 nM T99347 CQS0M7 24772040 IC50 > 10000 nM T99347 C5FTX6 24777576 EC50 = 980 nM T99347 C5RLE4 24777939 EC50 = 1080 nM T99347 CM0G3W 24782262 Ki = 195.2 nM T99347 C6N0OM 24782761 Ki = 434.7 nM T99347 C9Y1AN 24784504 IC50 = 1200 nM T99347 CASI47 24784989 IC50 = 2900 nM T99347 CQ3U2Z 24785223 IC50 = 230 nM T99347 CUZ1C3 24785482 IC50 = 250 nM T99347 CR9QJ8 24785549 Ki = 68.2 nM T99347 CZWY29 24785552 Ki = 103 nM T99347 CBF6J9 24815439 EC50 > 15848.93 nM T99347 CA02HI 24853384 IC50 = 7 nM T99347 C0XQA3 24884476 IC50 = 1220 nM T99347 CB9C4E 24965063 Ki = 9.8 nM T99347 CZXC58 24965064 Ki = 22 nM T99347 C0KXN2 25022596 IC50 = 0.7943 nM T99347 CQ1H5I 25101880 IC50 = 180 nM T99347 CJ82SE 25101881 IC50 = 360 nM T99347 C7CHW8 25102023 IC50 = 200 nM T99347 C13OIR 25145894 EC50 = 384 nM T99347 CI9EJ8 25145895 EC50 = 630 nM T99347 CSN89J 25167715 IC50 = 74 nM T99347 CG78YQ 25167856 IC50 = 43 nM T99347 CLI50W 25167857 IC50 = 27 nM T99347 CN0F4Z 25167988 IC50 = 21 nM T99347 CA8BN7 25168256 IC50 = 12 nM T99347 C74UXI 25168257 IC50 = 13 nM T99347 CS1AB2 25168520 Ki = 17 nM T99347 CH71MZ 25168801 IC50 = 25 nM T99347 CH06WV 25168930 Ki = 4.9 nM T99347 C16FZR 25168932 IC50 = 20 nM T99347 C16SYW 25169193 IC50 = 25 nM T99347 CPZG12 25169464 IC50 = 69 nM T99347 CS8GE1 25181642 Ki = 264.3 nM T99347 CGE8V0 25181656 Ki = 18.5 nM T99347 CZUP40 25181801 Ki = 20.4 nM T99347 C5AKX1 25181802 Ki = 3.3 nM T99347 C79LPB 25183668 Ki = 0.5 nM T99347 CHJY51 25183669 Ki = 11.9 nM T99347 CN8P7E 25183670 Ki = 0.3 nM T99347 CZC85B 25183673 Ki = 0.4 nM T99347 C0Q8BN 25183817 Ki = 18.4 nM T99347 CF46YL 25183819 Ki = 2.5 nM T99347 C89CXW 25183820 Ki = 24 nM T99347 CZ6N3X 25183826 Ki = 29.2 nM T99347 CO94PZ 25344457 Ki > 10000 nM T99347 CM3LG8 31565527 IC50 > 30000 nM T99347 CG8L3F 42765182 IC50 = 2400 nM T99347 CPID02 42765274 IC50 = 10000 nM T99347 C1KW3X 42765343 EC50 = 2700 nM T99347 C47HXB 42891592 EC50 = 1300 nM T99347 C7YN1F 42956962 EC50 = 3400 nM T99347 C2JI1Y 44089622 IC50 = 370 nM T99347 C5WR4B 44089674 IC50 = 2300 nM T99347 CUS97G 44089716 EC50 = 1200 nM T99347 CG01XT 44090476 IC50 = 630 nM T99347 CHQY08 44090528 IC50 = 690 nM T99347 CQY5F1 44091137 IC50 = 1100 nM T99347 C01RAS 44091218 EC50 = 1100 nM T99347 C0ZX4B 44091231 EC50 = 88 nM T99347 CN4B0R 44091484 IC50 = 680 nM T99347 C3P6RQ 44091531 IC50 = 1100 nM T99347 CRF28A 44091558 EC50 = 4800 nM T99347 C7TY5C 44091571 EC50 = 630 nM T99347 C2UQF8 44091572 EC50 = 1700 nM T99347 CT3RJ7 44091574 EC50 = 140 nM T99347 C1I9QM 44093855 IC50 = 3600 nM T99347 CERG28 44136108 IC50 = 10000 nM T99347 CC25MB 44136109 IC50 = 316.23 nM T99347 C9CZS7 44136507 IC50 = 125.89 nM T99347 CVK7F8 44136508 IC50 > 31622.78 nM T99347 CO0GC4 44157259 Ki = 2.7 nM T99347 CGA8B4 44157339 Ki = 11.4 nM T99347 CU5AB7 44158090 Ki = 3330 nM T99347 C4VZH3 44158331 Ki > 10000 nM T99347 CDR54S 44158332 Ki > 10000 nM T99347 CDO96T 44158334 Ki > 10000 nM T99347 CNF72Q 44190035 EC50 = 14 nM T99347 CVG97Y 44224177 IC50 = 840 nM T99347 C87KIW 44224178 IC50 = 9300 nM T99347 CBS17K 44224179 IC50 > 10000 nM T99347 C3WL6N 44230992 IC50 = 10 nM T99347 C09VPJ 44243470 IC50 = 19 nM T99347 CL13FV 44302605 IC50 > 300000 nM T99347 C03QML 44302608 IC50 > 300000 nM T99347 C2H6QV 44302609 IC50 > 300000 nM T99347 CP1QS5 44302686 IC50 > 300000 nM T99347 CR0JD5 44302687 IC50 = 99000 nM T99347 C0V9DN 44302818 IC50 > 300000 nM T99347 CDM1P2 44302819 IC50 > 300000 nM T99347 C1GV9Q 44302837 IC50 > 300000 nM T99347 C1FJU0 44302855 IC50 > 300000 nM T99347 C34AVQ 44302856 IC50 > 300000 nM T99347 CLF56U 44302896 IC50 > 300000 nM T99347 C9Y6QA 44302913 IC50 > 300000 nM T99347 CC7BN3 44302929 IC50 > 300000 nM T99347 CKL1M8 44302930 IC50 > 300000 nM T99347 C9U0NH 44302931 IC50 > 300000 nM T99347 CD5XY2 44302932 IC50 > 300000 nM T99347 C5ROF1 44322518 Ki > 10000000 nM T99347 C7E8SH 44322745 Ki = 1000000 nM T99347 CWV7F0 44322840 Ki > 100000 nM T99347 CGL0Z3 44322843 Ki > 1000000 nM T99347 C2SKJ1 44322921 Ki = 720 nM T99347 CR1OL6 44328753 IC50 > 100000 nM T99347 CUA80G 44328850 IC50 > 100000 nM T99347 C2SH0O 44329024 IC50 > 100000 nM T99347 CX0Y4F 44329029 IC50 = 5400 nM T99347 C76LOU 44329031 IC50 = 56100 nM T99347 CCV4N5 44329032 IC50 > 100000 nM T99347 CDP86T 44329033 IC50 > 100000 nM T99347 C9V5XC 44329042 IC50 > 100000 nM T99347 C6DC9V 44345143 IC50 = 19 nM T99347 C3U7JF 44389225 IC50 = 23 nM T99347 C94ZFX 44389261 IC50 = 3800 nM T99347 CHBP15 44389282 IC50 = 5084 nM T99347 C06RGT 44392945 IC50 = 2 nM T99347 CF6Y7L 44392951 IC50 = 4 nM T99347 C7XIO0 44392965 IC50 = 22 nM T99347 C1X7TD 44392969 IC50 = 3 nM T99347 CK78BW 44392972 IC50 = 29 nM T99347 C2IZF6 44392986 IC50 = 18 nM T99347 CUAP87 44395411 IC50 = 982 nM T99347 CC7W8F 44395412 IC50 = 251 nM T99347 CM2JG9 44395415 IC50 = 3000 nM T99347 CY38UL 44395430 IC50 = 497 nM T99347 CV5J6N 44395431 IC50 = 664 nM T99347 C6R2BN 44395437 IC50 = 2059 nM T99347 CX50JM 44395453 IC50 = 451 nM T99347 C1NOG9 44395459 IC50 = 335 nM T99347 CTU5A7 44395461 IC50 = 1467 nM T99347 C8Y6NP 44395489 IC50 = 445 nM T99347 C8FK9O 44395490 IC50 = 824 nM T99347 CM46YK 44395493 IC50 = 949 nM T99347 C27ICG 44395498 IC50 = 75 nM T99347 CW3GU1 44395504 IC50 = 271 nM T99347 CEI14T 44395505 IC50 = 287 nM T99347 C7A5XV 44395525 IC50 = 1171 nM T99347 CQW0B8 44395526 IC50 = 1546 nM T99347 CF50WY 44395531 IC50 = 120 nM T99347 CYN0B6 44395532 IC50 = 201 nM T99347 CU2F8G 44395543 IC50 = 575 nM T99347 C1JQ8S 44395544 IC50 = 806 nM T99347 CT3G5U 44395553 IC50 = 247 nM T99347 CR3F7L 44395559 IC50 = 337 nM T99347 COQ6N4 44395560 IC50 = 966 nM T99347 C86POR 44395563 IC50 = 108 nM T99347 C71SXJ 44395564 IC50 = 108 nM T99347 CZ7W5L 44395566 IC50 = 882 nM T99347 CRX18B 44395567 IC50 = 3000 nM T99347 CAJ7Q4 44395568 IC50 = 94 nM T99347 CLR0Q4 44395569 IC50 = 201 nM T99347 CBJ9R3 44395585 IC50 = 3000 nM T99347 C2L8NH 44395597 IC50 = 54 nM T99347 C5CJ6U 44395598 IC50 = 418 nM T99347 CAX8W2 44395599 IC50 = 217 nM T99347 CS7K3V 44395605 IC50 = 318 nM T99347 C9W1TG 44395609 IC50 = 223 nM T99347 CKZ3I6 44395613 IC50 = 418 nM T99347 CFG03J 44395622 IC50 = 30 nM T99347 CN2H0Y 44395630 IC50 = 316 nM T99347 C47MQD 44395631 IC50 = 342 nM T99347 CU6XY9 44395637 IC50 = 1000 nM T99347 C1VTG3 44395638 IC50 = 3000 nM T99347 C08HFT 44395640 IC50 = 150 nM T99347 C46TBK 44395641 IC50 = 151 nM T99347 C8Q9RO 44395644 IC50 = 359 nM T99347 C09NQP 44395645 IC50 = 389 nM T99347 CIZ60E 44395657 IC50 = 1458 nM T99347 CH09WZ 44395661 IC50 = 288 nM T99347 CW9XO4 44395665 IC50 = 312 nM T99347 CBY9F5 44395668 IC50 = 113 nM T99347 C53ABH 44395669 IC50 = 307 nM T99347 CXHM84 44395671 IC50 = 875 nM T99347 CCA52K 44395676 IC50 = 316 nM T99347 CH1Y8X 44395679 IC50 = 1577 nM T99347 CRP79D 44395684 IC50 = 376 nM T99347 C5E6SM 44398255 EC50 = 740 nM T99347 C1T6FL 44403551 IC50 = 12.6 nM T99347 C38UXS 44403552 IC50 = 2.6 nM T99347 CB53OS 44403559 IC50 = 35 nM T99347 CZAQ28 44403560 IC50 = 12 nM T99347 CGCH95 44403561 IC50 = 58 nM T99347 CG2OH1 44403566 IC50 = 8.2 nM T99347 CZI1N2 44403567 IC50 = 7.9 nM T99347 CMTK80 44403641 IC50 = 213 nM T99347 CO2D8P 44403647 IC50 = 22 nM T99347 CYG03F 44403648 IC50 = 16 nM T99347 C9I2HG 44403651 IC50 = 8.6 nM T99347 CSO48M 44403652 IC50 = 2.2 nM T99347 CO97KA 44403653 IC50 = 0.9 nM T99347 CJX0Z1 44403657 IC50 = 306 nM T99347 CWVR27 44403658 IC50 = 987 nM T99347 C62KFD 44404888 IC50 = 513 nM T99347 CA57ZI 44404889 IC50 = 243 nM T99347 C8ZX3V 44404893 IC50 = 267 nM T99347 CL1Q7X 44404926 IC50 = 1000 nM T99347 CXD85V 44404932 IC50 = 790 nM T99347 CQ2EP7 44404939 IC50 = 394 nM T99347 CND93U 44404946 IC50 = 36 nM T99347 CT6V1X 44407000 IC50 > 10000 nM T99347 CX31QU 44407032 IC50 > 10000 nM T99347 CMG2W6 44407071 IC50 > 10000 nM T99347 CFJ45E 44408211 IC50 > 10000 nM T99347 CX53RN 44408212 IC50 = 260 nM T99347 CV5H4B 44409632 Ki > 10000 nM T99347 CCO0P9 44409635 Ki = 1500 nM T99347 C2J6LR 44409636 Ki = 900 nM T99347 C72FIC 44409646 Ki = 160 nM T99347 C9JMN5 44409647 Ki = 28 nM T99347 C61KNG 44409671 Ki = 33 nM T99347 CZV02F 44409788 Ki = 48 nM T99347 C9V4RB 44409803 Ki = 17 nM T99347 C9LO4P 44409818 Ki = 70 nM T99347 C16KCN 44409819 Ki = 27 nM T99347 C3SA1B 44409828 Ki = 45 nM T99347 CQ4S6K 44409829 Ki > 3000 nM T99347 CFI57M 44409830 Ki = 44 nM T99347 CX40TQ 44409835 Ki = 51 nM T99347 C5BN2Y 44409875 Ki > 3000 nM T99347 C6MYA9 44409876 Ki = 18 nM T99347 CCI7U4 44409949 Ki = 27 nM T99347 C7C3VL 44410032 Ki = 4.7 nM T99347 C6RE9F 44410034 Ki = 6 nM T99347 CZ85AV 44410035 Ki = 3900 nM T99347 C5WP0Y 44410038 Ki = 11 nM T99347 CJ84BZ 44410400 IC50 > 10000 nM T99347 C7DXJ4 44410516 IC50 = 2370 nM T99347 CR9T5C 44410619 IC50 > 10000 nM T99347 CZYU46 44410647 IC50 > 10000 nM T99347 CH0X6R 44410649 IC50 > 3000 nM T99347 C6WNF2 44410650 IC50 > 10000 nM T99347 CC9NX8 44410672 IC50 > 10000 nM T99347 C6HQT1 44415851 IC50 > 10000 nM T99347 C98WYA 44415852 IC50 > 10000 nM T99347 CBZ80K 44415853 IC50 > 10000 nM T99347 C84UNW 44415865 IC50 > 10000 nM T99347 CC9L5P 44415866 IC50 > 10000 nM T99347 CO73DY 44415867 IC50 > 10000 nM T99347 CJDQ80 44415963 IC50 = 101 nM T99347 COJ36V 44415964 IC50 = 709 nM T99347 CEZ35Q 44415982 IC50 > 10000 nM T99347 C0D4RH 44415983 IC50 = 461 nM T99347 CC1J7P 44416001 IC50 > 10000 nM T99347 C4IMP1 44416002 IC50 = 2614 nM T99347 C1ET3W 44416003 IC50 > 10000 nM T99347 CF2O5C 44416005 IC50 = 306 nM T99347 CA9VD1 44416124 IC50 = 300 nM T99347 C6YQC3 44416142 IC50 = 7926 nM T99347 CL2WN6 44416143 IC50 > 10000 nM T99347 CO4J3C 44416193 IC50 > 3000 nM T99347 CMBQ83 44416254 IC50 = 1490 nM T99347 C7W0KG 44416271 IC50 = 825 nM T99347 C2PTH0 44416358 IC50 > 10000 nM T99347 CH8QG0 44416372 IC50 = 2490 nM T99347 C36JLH 44421618 IC50 > 100000 nM T99347 C4F0NS 44438457 Ki = 68 nM T99347 CPHX89 44438458 Ki > 10000 nM T99347 CXA35L 44438459 Ki = 397 nM T99347 CBN6P0 44438460 Ki = 2900 nM T99347 CRXN28 44438463 Ki = 3900 nM T99347 CCMI80 44438466 Ki > 10000 nM T99347 CMCJ80 44438468 Ki = 3900 nM T99347 C32SBE 44438470 Ki > 10000 nM T99347 CK4Q3M 44438471 Ki > 10000 nM T99347 CSE5H7 44438475 Ki = 2200 nM T99347 C5JW4C 44438477 Ki = 56 nM T99347 CKG59J 44438479 Ki = 327 nM T99347 C3WQ5E 44438482 Ki = 485 nM T99347 CO43SR 44438484 IC50 = 104 nM T99347 C2HBE4 44438486 Ki = 3900 nM T99347 CCY7Z9 44438491 Ki > 10000 nM T99347 C9DKN3 44438492 Ki = 3800 nM T99347 C4CTW5 44438495 Ki > 10000 nM T99347 C2FNS7 44438497 Ki = 251 nM T99347 C3RU2T 44438502 Ki = 250 nM T99347 CF3DH4 44438505 Ki = 1970 nM T99347 CAP72W 44438506 Ki = 3100 nM T99347 C89JMO 44438629 IC50 = 5 nM T99347 C3ZNV0 44438630 IC50 = 286 nM T99347 C0XWA3 44438631 IC50 = 39 nM T99347 CPE24T 44438632 IC50 = 26 nM T99347 CF3O2E 44440723 IC50 = 7300 nM T99347 CM9S3G 44440736 IC50 = 12400 nM T99347 CX7HD3 44441354 EC50 = 1500 nM T99347 C0F2DB 44441355 EC50 = 1400 nM T99347 CI45ZK 44441357 EC50 > 100000 nM T99347 CLC24K 44441361 EC50 = 720 nM T99347 C1FWH9 44441362 EC50 = 280 nM T99347 C9VHX8 44441363 EC50 > 100000 nM T99347 CR5WP0 44441365 EC50 > 100000 nM T99347 CF3CJ5 44441367 EC50 > 100000 nM T99347 CQ76HU 44441368 EC50 = 2200 nM T99347 C4L2RK 44441374 EC50 = 35000 nM T99347 C7Q6YE 44441376 EC50 > 100000 nM T99347 CTD58E 44441377 EC50 > 100000 nM T99347 C6QSM1 44441379 EC50 = 5700 nM T99347 CI10YE 44441381 EC50 > 100000 nM T99347 CT38KL 44441388 EC50 = 5700 nM T99347 C4MY9U 44441391 EC50 = 1900 nM T99347 C9QF3L 44441409 EC50 = 1700 nM T99347 CEHK42 44441410 EC50 = 4500 nM T99347 CN8RC6 44442420 IC50 > 100000 nM T99347 CJD2R3 44442421 IC50 = 100000 nM T99347 CS6HF7 44442422 IC50 > 100000 nM T99347 CE36NS 44442424 IC50 = 2800 nM T99347 CPXN04 44442425 IC50 = 3600 nM T99347 C0B5VU 44442426 IC50 > 100000 nM T99347 CKRV87 44442427 IC50 > 100000 nM T99347 CH4C8M 44442428 IC50 = 9500 nM T99347 CL4J2I 44442429 IC50 > 100000 nM T99347 C5FIC0 44442430 IC50 > 100000 nM T99347 CQ74SX 44442432 IC50 > 100000 nM T99347 C5F9EB 44442433 IC50 > 100000 nM T99347 C34NJZ 44442434 IC50 > 100000 nM T99347 CBEQ37 44442435 IC50 > 100000 nM T99347 CJ39IF 44442436 IC50 > 100000 nM T99347 C5P6AZ 44452891 IC50 = 100 nM T99347 C4P2FN 44452892 IC50 = 316.23 nM T99347 C8OZ2W 44452893 IC50 = 39.81 nM T99347 CSL59Z 44452895 IC50 = 398.11 nM T99347 C1EJW7 44452911 IC50 = 125.89 nM T99347 C4I7MR 44452913 IC50 = 3981.07 nM T99347 CXC9N3 44452914 IC50 = 1258.93 nM T99347 CYL3T6 44452917 IC50 = 630.96 nM T99347 CA31FW 44452939 IC50 = 251.19 nM T99347 C1D8WF 44452940 IC50 = 158.49 nM T99347 C9LE2S 44452943 IC50 = 199.53 nM T99347 CA73OY 44452966 IC50 = 10 nM T99347 CY0W9P 44452967 IC50 = 1258.93 nM T99347 C6DXS1 44452968 IC50 = 19.95 nM T99347 CB3TX7 44452969 IC50 = 12.59 nM T99347 CBAP39 44452995 IC50 = 125.89 nM T99347 CME7Y2 44452996 IC50 = 19.95 nM T99347 CANG89 44453018 IC50 = 158.49 nM T99347 CL6U4B 44453019 IC50 = 251.19 nM T99347 CFHS07 44453020 IC50 = 19.95 nM T99347 CT1IS2 44453023 IC50 = 50.12 nM T99347 CI35HL 44453044 IC50 = 199.53 nM T99347 CC28KP 44453045 IC50 = 50.12 nM T99347 C82HUB 44453046 IC50 = 1584.89 nM T99347 CBR40M 44453047 IC50 = 100 nM T99347 C4XW8G 44453071 IC50 = 501.19 nM T99347 C7DS0T 44453072 IC50 = 79.43 nM T99347 CJN5G1 44453073 IC50 = 7.943 nM T99347 C3LUT1 44453074 IC50 = 1584.89 nM T99347 C25CJO 44453075 IC50 = 316.23 nM T99347 CB21OU 44453141 IC50 = 19.95 nM T99347 C5PX0A 44453143 IC50 = 0.3981 nM T99347 CF8DS4 44453144 IC50 > 12589.25 nM T99347 CW3O9U 44453145 IC50 = 125.89 nM T99347 CZ5JC7 44453146 IC50 = 794.33 nM T99347 CW3EQ2 44453147 IC50 > 12589.25 nM T99347 C4O9LA 44453183 IC50 = 15.85 nM T99347 COD2I1 44453184 IC50 = 12.59 nM T99347 CQ2IO6 44453185 IC50 > 12589.25 nM T99347 C0LQY4 44453213 IC50 = 3.162 nM T99347 CPMF42 44453214 IC50 = 100 nM T99347 C7VN3B 44453215 IC50 = 25.12 nM T99347 C1VH5F 44453246 IC50 = 5011.87 nM T99347 C12LQM 44453247 IC50 = 316.23 nM T99347 CD9R8N 44453248 IC50 = 15.85 nM T99347 CO1K5J 44453249 IC50 = 1995.26 nM T99347 CXY3F5 44453250 IC50 = 63.1 nM T99347 C9IS8G 44453251 IC50 = 79.43 nM T99347 CZ9NO7 44453274 IC50 = 10000 nM T99347 CFTC02 44453277 IC50 > 12589.25 nM T99347 C7B0SY 44453278 IC50 = 158.49 nM T99347 CM3U4Y 44453279 IC50 > 12589.25 nM T99347 C7CJP3 44453307 IC50 = 10 nM T99347 C8PEH1 44453309 IC50 > 15848.93 nM T99347 C7J4VA 44453310 IC50 = 15.85 nM T99347 CBXC42 44453345 IC50 = 79.43 nM T99347 CYM9Z7 44453346 IC50 = 398.11 nM T99347 CF0G7O 44453347 IC50 = 100 nM T99347 CS3TM0 44453348 IC50 = 1.259 nM T99347 CIG03M 44453350 IC50 = 39.81 nM T99347 C1D0KV 44453384 IC50 > 3981.07 nM T99347 CHK4P8 44453385 IC50 > 15848.93 nM T99347 CCY12R 44453386 IC50 = 158.49 nM T99347 CY31SA 44453387 IC50 = 199.53 nM T99347 CL87VH 44453390 IC50 > 12589.25 nM T99347 CML3B0 44453391 IC50 = 1995.26 nM T99347 C2I7UY 44453420 IC50 = 316.23 nM T99347 C4NK1J 44453422 IC50 = 158.49 nM T99347 CN8VI2 44453423 IC50 = 501.19 nM T99347 CZ6AR4 44453453 IC50 = 125.89 nM T99347 CVIR06 44453454 IC50 > 12589.25 nM T99347 C7DT0S 44453455 IC50 = 316.23 nM T99347 CZ91PY 44453459 IC50 = 630.96 nM T99347 C3T4EV 44453482 IC50 = 794.33 nM T99347 CL9K6V 44453485 IC50 = 6.31 nM T99347 CX17MQ 44453486 IC50 > 12589.25 nM T99347 C72IFB 44453487 IC50 = 50.12 nM T99347 CN6W5D 44453488 IC50 = 10 nM T99347 CA7TG3 44453490 IC50 = 15.85 nM T99347 CFQ39N 44453492 IC50 = 0.3981 nM T99347 CD4JC0 44453494 IC50 = 2.512 nM T99347 CVJP38 44453515 IC50 = 50.12 nM T99347 CZTH17 44453516 IC50 = 63.1 nM T99347 C6XNM2 44453542 IC50 = 50.12 nM T99347 C4EWR5 44453543 IC50 = 501.19 nM T99347 CELT90 44453544 IC50 > 12589.25 nM T99347 CKD2Y7 44453546 IC50 > 15848.93 nM T99347 CWJ5G8 44453547 IC50 = 79.43 nM T99347 CFT89L 44453573 IC50 > 15848.93 nM T99347 C3Y5CJ 44453574 IC50 > 15848.93 nM T99347 CG1S0L 44453596 IC50 = 398.11 nM T99347 CX2M7G 44453598 IC50 > 15848.93 nM T99347 CE4U0K 44453599 IC50 > 15848.93 nM T99347 C4GWQ0 44453600 IC50 > 15848.93 nM T99347 CW47GH 44453601 IC50 > 15848.93 nM T99347 CGCT69 44453602 IC50 > 15848.93 nM T99347 CDOS16 44453603 IC50 = 100 nM T99347 CEZI59 44453604 IC50 = 1995.26 nM T99347 C15IFS 44453627 IC50 = 199.53 nM T99347 CXQ97M 44453628 IC50 = 3.162 nM T99347 C4W8OY 44453630 IC50 > 15848.93 nM T99347 CZ15DY 44453631 IC50 = 5011.87 nM T99347 CZG3T6 44569826 Ki > 300000 nM T99347 CJ28TF 44569827 Ki = 336000 nM T99347 CFZ64A 44569859 Ki = 293000 nM T99347 CUW74T 44569860 Ki > 300000 nM T99347 C2IKO1 44569861 Ki > 300000 nM T99347 CADV97 44569862 Ki > 1000000 nM T99347 CPC6B9 44574111 Ki = 0.9 nM T99347 C0DJ2Z 44588385 IC50 = 1000 nM T99347 CQ9IK3 44588386 IC50 = 1100 nM T99347 C8QXF5 44588425 IC50 = 1100 nM T99347 C2ZS9A 44588426 IC50 = 880 nM T99347 C58NLO 44588427 IC50 = 4000 nM T99347 CMEC89 44588428 IC50 = 8600 nM T99347 C1SBZ0 44588429 IC50 > 10000 nM T99347 CVKW41 44588460 IC50 = 8700 nM T99347 CTJA65 44588461 IC50 = 8300 nM T99347 CL24ZS 44588462 IC50 > 10000 nM T99347 CP5O4L 44588463 IC50 = 4300 nM T99347 CKTI06 44588464 IC50 = 170 nM T99347 CH4TG0 44593410 EC50 = 3300 nM T99347 CFAM64 45082292 EC50 = 19000 nM T99347 CZF26K 45265954 EC50 = 250 nM T99347 CAW5V1 45266964 EC50 = 46 nM T99347 CV4KU2 45268730 EC50 = 6600 nM T99347 CKGX75 45268733 EC50 = 140 nM T99347 CPTJ65 45269593 EC50 = 1600 nM T99347 CVE7A3 45270429 EC50 = 240 nM T99347 CKT7R8 45270430 EC50 = 990 nM T99347 CXL6A1 45271256 EC50 = 1200 nM T99347 C02EZW 45271257 EC50 = 180 nM T99347 C2WXM9 45271260 EC50 = 130 nM T99347 C5B8YR 45272146 EC50 = 510 nM T99347 CXLW08 45272148 EC50 = 1200 nM T99347 C4FAS1 45272149 EC50 = 280 nM T99347 CI6NA2 45486778 IC50 > 10000 nM T99347 C0N2HC 45486816 IC50 = 6600 nM T99347 CTL13I 46226029 IC50 = 95 nM T99347 CO70UN 46226030 IC50 = 1600 nM T99347 CF6YI1 46226033 IC50 > 10000 nM T99347 CZLJ19 46226035 IC50 = 2300 nM T99347 C7MF8K 46226036 IC50 > 10000 nM T99347 CN7T4C 46226039 IC50 > 10000 nM T99347 C1FVX9 46226040 IC50 = 2100 nM T99347 CRM1Z0 46226041 IC50 > 10000 nM T99347 CR9M3F 46226042 IC50 = 720 nM T99347 CT78ZO 46226043 IC50 = 980 nM T99347 CE04OM 46226044 IC50 > 10000 nM T99347 C2K3UR 46226045 IC50 > 10000 nM T99347 C45ZQO 46226046 IC50 > 10000 nM T99347 C31PAF 46700737 EC50 > 10000 nM T99347 C15XWL 46742816 EC50 = 117.49 nM T99347 CGS4F2 46836713 EC50 > 10000 nM T99347 C13FOU 46853594 IC50 = 16 nM T99347 CY5Q8L 46886118 IC50 > 3000 nM T99347 C1B5XO 46886119 IC50 > 3000 nM T99347 C4YD2C 46886120 IC50 > 3000 nM T99347 CM9KV2 46886135 IC50 > 3000 nM T99347 CR1O4K 46886136 IC50 > 3000 nM T99347 CYO8Z9 46886137 IC50 > 3000 nM T99347 CJ57LM 46886138 IC50 > 3000 nM T99347 CAF9X1 46886139 IC50 > 3000 nM T99347 CG6W8P 46886140 IC50 > 3000 nM T99347 C6SYU4 46886169 IC50 > 3000 nM T99347 CJ0TA9 46912224 IC50 = 290 nM T99347 CR53OV 46931800 IC50 = 2600 nM T99347 CW6AE9 46932105 IC50 = 153 nM T99347 C1QBU6 46932196 IC50 = 346 nM T99347 CPU4F7 46932381 IC50 = 640 nM T99347 CR2ON6 46932384 IC50 = 54 nM T99347 C6XD7O 46932857 IC50 = 60 nM T99347 CUF9A1 49782363 IC50 = 1200 nM T99347 CWQH64 49782364 IC50 = 110 nM T99347 C8TYP5 49782369 IC50 = 330 nM T99347 C51QXZ 49782573 IC50 = 28 nM T99347 CC7T4M 49782804 IC50 = 57 nM T99347 CV6F9U 49799828 IC50 > 300000 nM T99347 C1N4ID 49832807 IC50 = 560 nM T99347 CH2LC7 50914184 EC50 = 17.38 nM T99347 CU05LX 51003579 EC50 = 15.8 nM T99347 CH9MG2 51003580 EC50 = 30.2 nM T99347 CWE2O4 51033723 Ki = 2.4 nM T99347 C0L2SP 51036108 EC50 > 30000 nM T99347 CAU6D5 51036701 EC50 > 30000 nM T99347 CBI3A0 51036916 EC50 > 30000 nM T99347 C3GQ8O 51037131 EC50 > 30000 nM T99347 CV86OW 51049976 EC50 = 6.1 nM T99347 C2EBK3 51346800 EC50 = 5.9 nM T99347 C5U4YC 51346801 EC50 = 12 nM T99347 CY2WM8 52941509 EC50 = 390 nM T99347 CAJ9G5 52941568 EC50 > 10600 nM T99347 CG13KV 52942503 EC50 = 290 nM T99347 CY6H3K 52942601 EC50 = 350 nM T99347 C62FZO 52942704 EC50 = 240 nM T99347 CH1KM8 52942917 EC50 = 2100 nM T99347 C2XAR7 52943881 EC50 = 570 nM T99347 CQEO36 52943923 EC50 = 680 nM T99347 CK9N3O 52944770 EC50 = 8500 nM T99347 C8IPL7 52944881 EC50 = 5200 nM T99347 C8ECF1 52946009 EC50 > 25000 nM T99347 CI7Q9U 52946010 EC50 = 7100 nM T99347 CRS3T0 52946160 EC50 > 310 nM T99347 C6UM8P 52946222 EC50 = 6700 nM T99347 CD0Q4E 52946360 EC50 = 4200 nM T99347 C6P1MR 52946490 EC50 = 18000 nM T99347 CI85AK 52947238 EC50 > 25000 nM T99347 CGB12H 52947293 EC50 > 25000 nM T99347 CZ4DY9 52947518 EC50 = 600 nM T99347 C5H0KT 52947687 EC50 > 25000 nM T99347 CLZK95 52948447 EC50 = 5300 nM T99347 CA59IY 52948559 EC50 = 2800 nM T99347 C3X9AC 52948609 EC50 = 210 nM T99347 CA4WT3 52948680 IC50 = 129 nM T99347 CGCQ87 52948764 EC50 > 25000 nM T99347 CCO51I 52948810 EC50 = 370 nM T99347 CM9KC2 52948843 EC50 = 800 nM T99347 COR01F 52950067 EC50 = 6600 nM T99347 CKF3E8 53101051 IC50 = 770 nM T99347 CN1HU8 53235518 EC50 = 33 nM T99347 CY58NO 53240406 EC50 > 25000 nM T99347 CGV09X 53246019 EC50 = 112 nM T99347 C76AVE 53246020 EC50 = 2.4 nM T99347 C6SUW0 53246141 EC50 = 119 nM T99347 COV78P 53246490 EC50 = 1122.02 nM T99347 CB2W5G 53246601 EC50 = 851 nM T99347 CB0L9V 53246602 EC50 = 2290.87 nM T99347 CD25RT 53246605 EC50 = 739 nM T99347 CYUT81 53246607 EC50 = 95.5 nM T99347 C7B6YK 53246852 EC50 = 1737.8 nM T99347 C1MO0U 53246971 EC50 = 75.86 nM T99347 CA2L0H 53246975 EC50 = 66 nM T99347 CD2KS9 53246977 EC50 = 549.54 nM T99347 CVY36W 53247219 EC50 = 250 nM T99347 C2U0HG 53247224 EC50 = 1445.44 nM T99347 CVDI42 53247225 EC50 = 1019 nM T99347 C3DXS9 53247347 EC50 = 616.6 nM T99347 CZO7S9 53247348 EC50 = 1759 nM T99347 C8Q2AT 53247349 EC50 = 2690 nM T99347 C1J5WR 53247350 EC50 = 791 nM T99347 CFU9Y7 53247471 EC50 = 691.83 nM T99347 CZAK68 53247590 EC50 = 1202.26 nM T99347 C04LVW 53248876 EC50 = 5.9 nM T99347 CS25OY 53248877 EC50 = 239 nM T99347 CEP97G 53248878 IC50 = 776 nM T99347 CJ1S3D 53248879 IC50 = 5.7 nM T99347 C68AZB 53316663 IC50 = 3162.28 nM T99347 CS7T6M 53316664 IC50 = 12.59 nM T99347 C8UC4Y 53316688 IC50 = 39.81 nM T99347 CKOF26 53317110 EC50 = 53.2 nM T99347 CXBA68 53317111 EC50 > 25000 nM T99347 CXRP23 53317120 EC50 = 741.31 nM T99347 C3TSV6 53317121 EC50 = 204.17 nM T99347 C5CBV7 53317122 EC50 = 457.09 nM T99347 C3WU1S 53317123 EC50 = 602.56 nM T99347 C5LFQ2 53317271 EC50 = 180 nM T99347 CSC40L 53317272 EC50 = 150 nM T99347 C7ZO2S 53317273 EC50 > 10000 nM T99347 C3IQ6Z 53317437 EC50 = 270 nM T99347 CC8P5R 53317662 EC50 = 850 nM T99347 C1C2QH 53317970 IC50 = 10 nM T99347 CK47PZ 53317971 IC50 > 31622.78 nM T99347 CFT4M2 53318399 EC50 = 112.2 nM T99347 CN03BI 53318400 EC50 = 20.3 nM T99347 CNFA87 53318409 EC50 = 257.04 nM T99347 CT19UJ 53318410 EC50 = 524.8 nM T99347 CWK16Q 53318411 EC50 = 453.6 nM T99347 C9A3OP 53318558 EC50 = 160 nM T99347 CA8WS0 53318559 EC50 = 3600 nM T99347 C6FO3A 53318766 IC50 = 130 nM T99347 C92AXM 53318843 EC50 = 11.48 nM T99347 CL86OX 53319313 IC50 = 39.81 nM T99347 C8M5HI 53319314 IC50 = 39.81 nM T99347 CRP4M3 53319730 EC50 = 512.86 nM T99347 CM9DX3 53319731 EC50 = 562.34 nM T99347 CMR07F 53319732 EC50 = 307.8 nM T99347 CWI2Y6 53319739 EC50 = 295.1 nM T99347 CTS1F0 53319740 EC50 = 371.5 nM T99347 C3H9KU 53319741 EC50 = 831.76 nM T99347 CE89JI 53319877 EC50 = 54 nM T99347 CLY07W 53319878 EC50 = 56 nM T99347 CG4HS9 53319936 IC50 = 660 nM T99347 CW47QC 53319937 EC50 = 870 nM T99347 CV8G4K 53319938 EC50 = 5700 nM T99347 C3TB1J 53319939 EC50 = 170 nM T99347 CA1D0U 53320114 EC50 = 56.23 nM T99347 C8Y5NX 53320294 EC50 = 12.3 nM T99347 CKH4V8 53320613 IC50 = 63.1 nM T99347 C4JGA7 53320614 IC50 = 5011.87 nM T99347 CO75JQ 53320615 IC50 = 7.943 nM T99347 CD8G9Z 53321027 EC50 = 588.8 nM T99347 CMLC83 53321035 EC50 = 239.88 nM T99347 CR9EC0 53321036 EC50 = 60.26 nM T99347 CJWU45 53321182 EC50 = 3400 nM T99347 C64PBY 53321183 EC50 = 470 nM T99347 CE0N6S 53321242 EC50 = 350 nM T99347 C0TWY2 53321433 IC50 = 100 nM T99347 C2XZ5L 53321504 IC50 = 39.81 nM T99347 CTY26K 53321916 IC50 = 2511.89 nM T99347 C2D9GX 53321917 IC50 > 31622.78 nM T99347 CAS97H 53322366 EC50 = 181.97 nM T99347 C5TGB9 53322367 EC50 = 213.8 nM T99347 CB3Q0C 53322380 EC50 = 61.66 nM T99347 CKZ0C3 53322381 EC50 = 776.2 nM T99347 CW36CH 53322382 EC50 = 29.51 nM T99347 C4QF6V 53322457 EC50 = 900 nM T99347 C6TXY4 53322501 EC50 = 96 nM T99347 CO63CY 53322502 EC50 = 3700 nM T99347 CZ01WI 53323262 IC50 = 50.12 nM T99347 CIX93J 53323263 IC50 = 12.59 nM T99347 C6W2PB 53323727 EC50 = 29.51 nM T99347 C8L0FU 53323728 EC50 = 29.5 nM T99347 C12ZPO 53323736 EC50 = 208.9 nM T99347 C4A3YO 53323737 EC50 = 572.1 nM T99347 CO78WE 53323738 EC50 = 107.15 nM T99347 C8QTP6 53323739 EC50 = 154.88 nM T99347 CQOZ20 53323740 EC50 = 475 nM T99347 CO31KB 53323741 EC50 = 707.95 nM T99347 CU56RP 53323852 EC50 = 170 nM T99347 CX85IQ 53323908 EC50 = 35 nM T99347 CQ58TY 53324080 IC50 = 110 nM T99347 COY9K4 53325005 EC50 = 37.15 nM T99347 CL7T2A 53325124 EC50 = 250 nM T99347 C30ZGK 53325125 EC50 = 550 nM T99347 CC3DG5 53325126 EC50 = 4000 nM T99347 C6YGC7 53325127 EC50 = 610 nM T99347 CG4DV0 53325128 EC50 = 260 nM T99347 C30SHG 53325129 EC50 = 4900 nM T99347 C60TDV 53325186 EC50 = 66 nM T99347 CN27IK 53325298 EC50 > 10000 nM T99347 CP38XD 53325301 EC50 = 160 nM T99347 C5Y4EL 53325366 IC50 = 110 nM T99347 C6A9CQ 53325367 IC50 > 500 nM T99347 C43CVB 53325597 IC50 = 501.19 nM T99347 CK2DT1 53325624 EC50 = 200 nM T99347 CNR98D 53325898 IC50 = 10 nM T99347 CUH1F3 53325899 IC50 = 63.1 nM T99347 C0AUX4 53326305 EC50 = 691.83 nM T99347 CA5HY9 53326432 EC50 = 130 nM T99347 C0Z7JS 53326433 EC50 = 290 nM T99347 CLWV18 53326573 IC50 = 170 nM T99347 CIH1R8 53326844 EC50 = 107.15 nM T99347 CZ03BQ 54579958 IC50 > 3000 nM T99347 CVM2Z7 54579959 IC50 > 3000 nM T99347 COLN14 54580485 IC50 > 3000 nM T99347 CUFW72 54580598 IC50 = 22 nM T99347 CD5PG9 54580599 EC50 = 393 nM T99347 C8PN2E 54580600 EC50 = 12 nM T99347 CS4E9H 54580610 IC50 = 9300 nM T99347 CGO7T3 54580611 IC50 > 10000 nM T99347 CKG7T0 54580614 EC50 = 1500 nM T99347 CE0N3K 54580616 EC50 = 1400 nM T99347 C29NCQ 54580617 EC50 = 460 nM T99347 CZB36I 54580944 IC50 = 1180 nM T99347 C5O1LV 54580945 IC50 > 3000 nM T99347 CHFO58 54580946 IC50 > 3000 nM T99347 C3ST8U 54580947 IC50 > 3000 nM T99347 C1VR9A 54580948 IC50 > 3000 nM T99347 CE3VP1 54581505 IC50 > 3000 nM T99347 CN1M2A 54581607 EC50 = 62 nM T99347 C16UVZ 54581608 IC50 = 184 nM T99347 CXWQ54 54581609 Ki = 23150 nM T99347 CK90MI 54581620 IC50 = 2600 nM T99347 C0Z1HP 54581622 EC50 = 10000 nM T99347 C1OAP5 54581625 IC50 = 900 nM T99347 CIHC67 54582001 IC50 = 820 nM T99347 CCR0O3 54582002 IC50 > 3000 nM T99347 C2V1FR 54582003 IC50 > 3000 nM T99347 CSF8T1 54582004 IC50 > 3000 nM T99347 C0O6PC 54582005 IC50 > 3000 nM T99347 CYN49G 54582006 IC50 > 3000 nM T99347 CT6VC7 54582031 IC50 = 2350 nM T99347 CB8K2V 54582032 EC50 = 7600 nM T99347 CY9XF3 54582494 IC50 > 3000 nM T99347 CDK3M9 54582595 EC50 > 10000 nM T99347 CBMK01 54582596 IC50 = 30 nM T99347 C6BJ5X 54582597 IC50 = 810 nM T99347 CO7PM1 54582598 IC50 = 2517 nM T99347 CG34SP 54582599 IC50 = 111 nM T99347 CZ1TW4 54582600 IC50 = 27 nM T99347 CU0O7P 54582601 IC50 = 45 nM T99347 CTV6K7 54582602 EC50 = 7.5 nM T99347 C9PA3R 54582603 EC50 = 33 nM T99347 C7PO4M 54582604 EC50 = 462 nM T99347 C0RZJ9 54582615 IC50 = 4700 nM T99347 C48VIL 54582619 IC50 = 280 nM T99347 C04JGT 54582620 EC50 = 80 nM T99347 C53LYP 54582621 EC50 = 3500 nM T99347 C81WKP 54582622 IC50 = 730 nM T99347 C8DH7O 54582623 IC50 = 10000 nM T99347 C4CB9V 54582624 EC50 = 23000 nM T99347 CA6NZ2 54582941 IC50 > 30000 nM T99347 CM6QA5 54582942 IC50 > 3000 nM T99347 C19GTC 54582943 IC50 > 3000 nM T99347 CCY49K 54582944 IC50 > 3000 nM T99347 CWMT03 54582945 IC50 > 3000 nM T99347 CZ17AI 54582946 IC50 > 3000 nM T99347 CPZ83T 54583474 IC50 > 3000 nM T99347 CWUG79 54583563 IC50 = 451 nM T99347 CZV60O 54583564 IC50 = 4.8 nM T99347 CQIV04 54583565 EC50 = 1012 nM T99347 CN5O0I 54583570 IC50 = 3500 nM T99347 C9JY5Z 54583571 EC50 = 2600 nM T99347 CVGZ59 54583572 EC50 = 3600 nM T99347 CD8WI5 54583575 EC50 = 310 nM T99347 C4X1WI 54583713 IC50 = 10000 nM T99347 C2LT4E 54583940 IC50 = 5020 nM T99347 C0GSX1 54583941 IC50 > 30000 nM T99347 COAT86 54583942 IC50 > 3000 nM T99347 CTG4X9 54583943 IC50 > 3000 nM T99347 CZ5K2Y 54584442 IC50 > 3000 nM T99347 CXP59T 54584443 IC50 > 3000 nM T99347 CDW9T7 54584540 IC50 = 2.9 nM T99347 CMG93H 54584541 IC50 = 916 nM T99347 CP0NM6 54584542 IC50 = 4228 nM T99347 CXA7L5 54584543 EC50 = 979 nM T99347 CX26QC 54584544 EC50 = 748 nM T99347 CSMZ26 54584545 Ki = 27150 nM T99347 CES04A 54584546 IC50 = 518 nM T99347 C2XSG0 54584558 EC50 = 1000 nM T99347 CEK29H 54584559 EC50 = 3700 nM T99347 C9QWU4 54584560 EC50 = 10000 nM T99347 CF7XP3 54584561 EC50 = 530 nM T99347 CQ8BM3 54584565 EC50 = 600 nM T99347 C2KDJ8 54584566 EC50 = 2900 nM T99347 CQ98YR 54584567 EC50 = 2900 nM T99347 CME8Y2 54584583 EC50 = 13 nM T99347 CA6GY7 54584886 IC50 = 5240 nM T99347 C23PDM 54584887 IC50 > 3000 nM T99347 C8PW4R 54584888 IC50 > 3000 nM T99347 CY3P6J 54584889 IC50 > 3000 nM T99347 CB5MH3 54584890 IC50 > 3000 nM T99347 CSBE97 54584891 IC50 > 3000 nM T99347 CD26YU 54584892 IC50 > 3000 nM T99347 C3NC5O 54584919 EC50 = 6100 nM T99347 C6D9YF 54585403 IC50 > 3000 nM T99347 C5CBA9 54585404 IC50 > 3000 nM T99347 CR5K0W 54585405 IC50 > 3000 nM T99347 CB5Z9Y 54585406 IC50 > 3000 nM T99347 C57SJG 54585486 Ki = 15000 nM T99347 CUF9X3 54585487 IC50 = 293 nM T99347 C1R6BP 54585488 IC50 = 706 nM T99347 C16XMD 54585489 EC50 = 4816 nM T99347 CI8W3P 54585490 IC50 = 199 nM T99347 CB8JW5 54585491 EC50 = 171 nM T99347 C68RVS 54585492 Ki > 32000 nM T99347 CEUQ93 54585502 IC50 = 10000 nM T99347 CZ13FY 54585503 IC50 = 10000 nM T99347 C7G0QL 54585849 IC50 > 10000 nM T99347 CS1X5M 54585850 IC50 > 3000 nM T99347 C93WBA 54585851 IC50 > 3000 nM T99347 CFM8Q2 54585852 IC50 > 3000 nM T99347 CL4V8K 54585881 EC50 = 6500 nM T99347 C6WK1O 54586361 IC50 > 3000 nM T99347 CHU13F 54586362 IC50 > 3000 nM T99347 CE3X5Z 54586363 IC50 > 3000 nM T99347 CV29ZU 54586459 Ki = 19550 nM T99347 C2QYG3 54586460 EC50 = 36 nM T99347 C6NTE7 54586470 IC50 = 2400 nM T99347 CTR5W0 54586472 EC50 = 430 nM T99347 CG07AJ 54586473 EC50 = 7000 nM T99347 CDGO98 54586478 EC50 = 700 nM T99347 CI7WZ0 54586814 IC50 > 10000 nM T99347 C5BU8V 54586815 IC50 > 10000 nM T99347 C34IBD 54586816 IC50 > 10000 nM T99347 CF94LX 54586817 IC50 > 3000 nM T99347 CLPR07 54586818 IC50 > 3000 nM T99347 CILU43 54587386 IC50 > 3000 nM T99347 C21WLS 54587482 IC50 = 227 nM T99347 CA51OJ 54587483 IC50 = 1401 nM T99347 CH3OX8 54587484 IC50 = 352 nM T99347 CX1P8R 54587485 Ki = 27380 nM T99347 CXQI21 54587486 EC50 = 40 nM T99347 CX2H0W 54587487 EC50 = 466 nM T99347 C3P1GY 54587488 EC50 = 924 nM T99347 C7JRX4 54587489 EC50 = 387 nM T99347 CM4NS6 54587499 IC50 = 9900 nM T99347 C4Q6LE 54587500 IC50 = 700 nM T99347 CP8E3H 54587505 IC50 = 10000 nM T99347 CQSG40 54587506 IC50 = 4700 nM T99347 C1DL9H 54596257 IC50 = 0.79 nM T99347 CJRG27 54761054 EC50 > 30000 nM T99347 C8P1UJ 56659585 IC50 = 120 nM T99347 CA5V6M 56660085 IC50 = 2 nM T99347 CVO41Q 56660086 IC50 = 140 nM T99347 CGZ98M 56660087 IC50 = 8 nM T99347 CF8H5C 56660088 IC50 = 320 nM T99347 C0B7ZR 56663548 IC50 = 14 nM T99347 C8F1JC 56663549 IC50 = 140 nM T99347 C4BYF5 56663550 IC50 = 1900 nM T99347 CNP0T8 56663551 IC50 = 10000 nM T99347 C3RNC5 56663552 IC50 = 8 nM T99347 CG78SU 56663553 IC50 = 680 nM T99347 C23QYO 56663554 IC50 = 120 nM T99347 CI06EK 56663555 IC50 = 370 nM T99347 C65FOQ 56666997 IC50 = 23 nM T99347 CFGC12 56666998 IC50 = 10 nM T99347 C2F5OL 56666999 IC50 = 84 nM T99347 CVL59O 56667000 IC50 = 68 nM T99347 CUS89F 56670439 IC50 = 3 nM T99347 CHZB96 56670440 IC50 = 11 nM T99347 C2JH0G 56670441 IC50 = 120 nM T99347 CDRH30 56673923 IC50 = 5 nM T99347 CO6V5I 56673924 IC50 = 9 nM T99347 C7REH6 56673925 IC50 = 2400 nM T99347 CM4R9C 56673926 IC50 = 30 nM T99347 C4D2NA 56673927 IC50 = 80 nM T99347 CQI04X 56673928 IC50 = 320 nM T99347 CIWQ23 56673929 Ki = 130 nM T99347 CINW83 56677263 IC50 = 110 nM T99347 CB4M2U 56677264 Ki = 360 nM T99347 C1TK6P 56677265 IC50 = 2000 nM T99347 C8DU9K 56677266 IC50 = 74 nM T99347 CF3LG9 56680564 IC50 = 74 nM T99347 CGF6X8 56680565 IC50 = 94 nM T99347 CXZ97B 56683901 IC50 = 8 nM T99347 CH2QA1 56683902 IC50 = 41 nM T99347 CBZA50 56683903 IC50 = 390 nM T99347 C5A0TB 56941774 EC50 = 290 nM T99347 CP98VZ 56941777 EC50 = 1400 nM T99347 C3DP5Z 56962486 IC50 = 68.4 nM T99347 CTG79J 56963567 IC50 = 27.8 nM T99347 CY3B1Z 57330204 Ki = 1.6 nM T99347 COZ7L2 57388814 IC50 = 452 nM T99347 CG7CH6 57388815 IC50 = 4710 nM T99347 CA9CL8 57388816 IC50 = 2230 nM T99347 C3MOX5 57388817 IC50 = 120 nM T99347 C35JAV 57388818 IC50 = 722 nM T99347 CR87KW 57388819 IC50 = 272 nM T99347 CN83ZO 57388895 IC50 = 34.3 nM T99347 CA14YX 57388896 IC50 = 6160 nM T99347 C08OQJ 57388899 IC50 = 83.1 nM T99347 CI0AM2 57388978 IC50 = 43.2 nM T99347 CUOT05 57388979 IC50 = 111 nM T99347 CA7Q2X 57388981 IC50 = 1120 nM T99347 CY5S1I 57389059 IC50 = 245 nM T99347 CN79LA 57389060 IC50 = 493 nM T99347 CD9B7X 57389063 IC50 = 1040 nM T99347 C7WYD8 57389158 IC50 = 125 nM T99347 COMI92 57389235 IC50 = 1130 nM T99347 CDQE09 57389238 IC50 = 721 nM T99347 CB1HF7 57389241 IC50 = 157 nM T99347 CWK1D4 57404255 IC50 = 158 nM T99347 C6XA7G 57405264 EC50 = 370 nM T99347 CU76EW 57410027 EC50 = 300 nM T99347 CSU73H 57410141 EC50 = 3980 nM T99347 CR2TY0 57411802 EC50 = 100 nM T99347 CSH09Y 57411803 EC50 = 2340 nM T99347 CC8N9R 57559280 IC50 = 10000 nM T99347 CLUD90 57559287 IC50 = 10000 nM T99347 CZ6IE0 57559301 IC50 = 10000 nM T99347 CL0R2Q 57559313 IC50 = 1000 nM T99347 CVN1K2 57559437 IC50 = 10000 nM T99347 C0KGQ3 57559476 IC50 = 10000 nM T99347 CWTH50 57559504 IC50 = 10000 nM T99347 CZWP49 57559572 IC50 = 10000 nM T99347 CNBR74 57559597 IC50 = 10000 nM T99347 C4Z7LT 57559648 IC50 = 10000 nM T99347 CP16EG 57574885 Ki = 194 nM T99347 CY6O7G 57574904 Ki = 64.2 nM T99347 CAS3O2 57574912 Ki > 1000 nM T99347 CAQ71K 57574919 Ki = 15.8 nM T99347 CW4Y9L 57574921 Ki = 92 nM T99347 C8HYG7 57574929 Ki = 456 nM T99347 C12HQA 57574930 Ki = 122 nM T99347 C46ITO 57574931 Ki > 1000 nM T99347 CASM07 57574933 Ki = 67.3 nM T99347 C6STI7 57574945 Ki = 258 nM T99347 CZCK85 57574952 Ki = 415 nM T99347 CM1EK8 57574953 Ki = 2.9 nM T99347 CX4F6L 57574973 Ki = 40 nM T99347 CY5D1K 57574980 Ki = 2.9 nM T99347 C9CD2Y 57574990 Ki = 4.8 nM T99347 C3XGL6 57574995 Ki = 0.7 nM T99347 CR7K1C 57575007 Ki = 4.3 nM T99347 CG93BU 57575012 Ki = 11.3 nM T99347 CPE25J 57575026 Ki = 18.2 nM T99347 C0DR6M 57575029 Ki = 178 nM T99347 CEZ9T2 57575036 Ki = 399 nM T99347 C30NGS 57575054 Ki = 48.2 nM T99347 CM53TE 57577087 IC50 = 94 nM T99347 CVO9M5 57577106 IC50 = 25 nM T99347 C34TUB 57577121 IC50 = 22 nM T99347 CRJ02N 57577235 IC50 = 35 nM T99347 C7ORF4 57881625 IC50 = 10000 nM T99347 CTY0F2 57881665 IC50 = 200 nM T99347 C6MJB8 57908398 IC50 = 29 nM T99347 C1K3TI 57908399 IC50 = 36 nM T99347 C9UK4O 57908400 IC50 = 54 nM T99347 C4YVT6 57908404 IC50 = 45 nM T99347 C6P7NH 57927756 Ki = 55.6 nM T99347 C8N4UB 60096231 IC50 > 12500 nM T99347 C2D3HQ 60168069 IC50 = 14 nM T99347 CY04QB 60210882 EC50 = 4500 nM T99347 CV4UR6 60210898 EC50 > 10000 nM T99347 CS4AC9 60210916 EC50 > 10000 nM T99347 C6Q1US 66553219 IC50 = 1505 nM T99347 CDV0S7 66557172 IC50 = 54 nM T99347 CZF76R 66608383 EC50 = 239.88 nM T99347 CB4D1J 66608640 EC50 = 220 nM T99347 CR5Z4W 66608716 EC50 = 616.6 nM T99347 CGH3V0 66609011 EC50 = 139 nM T99347 CVHE21 66609033 EC50 = 640 nM T99347 CN5U0B 66609115 EC50 = 290 nM T99347 CSM1I0 66609338 EC50 = 150 nM T99347 CBLM26 66609382 EC50 = 660 nM T99347 C5O7YL 66609653 EC50 = 510 nM T99347 CNX90R 66609770 EC50 = 1200 nM T99347 C6RK5X 66613256 EC50 > 10000 nM T99347 C4I9TR 66613289 EC50 = 230 nM T99347 CYOU10 66613304 EC50 = 290 nM T99347 C9DTE1 66613308 EC50 > 10000 nM T99347 CF6LJ9 66613404 EC50 = 2454.71 nM T99347 CUP41L 66613450 EC50 = 546 nM T99347 C7FD2P 66613497 EC50 = 1700 nM T99347 C4PU9N 67056056 EC50 > 30000 nM T99347 C4RD2I 67179855 IC50 > 12500 nM T99347 CR84XZ 67180972 IC50 = 6650 nM T99347 C4NG6L 67181122 IC50 = 19 nM T99347 C71SCP 67181213 IC50 > 12500 nM T99347 CJ5G2L 67181693 IC50 > 12500 nM T99347 CFM52I 67182239 IC50 = 730 nM T99347 CG0LC2 67182345 IC50 = 159 nM T99347 CBX67G 67246999 EC50 = 1195 nM T99347 CW7BI6 67424364 IC50 = 39 nM T99347 CA9LV5 67424813 IC50 = 62 nM T99347 CC1HY4 67425269 IC50 = 30 nM T99347 C6M1FY 67425323 IC50 = 20 nM T99347 C4LO1P 67425408 IC50 = 81 nM T99347 C5JQ0F 67425734 IC50 = 45 nM T99347 CYL12Q 67510438 EC50 = 30.7 nM T99347 CYB12X 67973635 EC50 = 186.21 nM T99347 C03HIJ 67973779 EC50 = 489.78 nM T99347 CU89OF 67973795 EC50 = 158.49 nM T99347 CAS0X1 67973817 EC50 = 87 nM T99347 CLN87E 67973847 EC50 = 2089.3 nM T99347 CRS94B 67973913 EC50 = 70.79 nM T99347 C8B2QK 67974041 EC50 = 110 nM T99347 C9VUK7 67974056 EC50 > 30000 nM T99347 CJ4HA6 67974346 EC50 = 100 nM T99347 CX2I8F 67974348 EC50 = 616.6 nM T99347 C5K7QG 67974411 EC50 = 125.89 nM T99347 CC54XA 67974464 EC50 = 125.89 nM T99347 C0OZR7 67974471 EC50 = 758.58 nM T99347 CQ49LN 67974482 EC50 = 2089.3 nM T99347 C7HQ9Y 67974497 EC50 = 758.58 nM T99347 C75YSP 67974644 EC50 = 64.57 nM T99347 C3A2KP 67974705 EC50 = 147.91 nM T99347 CQLT10 67975734 EC50 = 100 nM T99347 CRC8N6 67975736 EC50 = 7940 nM T99347 CI1Y4R 67976002 EC50 = 690 nM T99347 CE3D6S 67976023 EC50 = 1230 nM T99347 CN29JR 67976044 EC50 = 7760 nM T99347 C5U9QX 69081596 EC50 = 0.8 nM T99347 CQ1MU4 69081973 Ki = 8.9 nM T99347 CC7G3J 69082917 EC50 = 0.6 nM T99347 CSA4R9 69083336 Ki = 6.5 nM T99347 CLV7Q3 69083418 Ki = 13 nM T99347 CKU4M1 69083983 EC50 = 0.9 nM T99347 CPCH65 69084420 EC50 = 6 nM T99347 CN3F8A 69084898 Ki = 0.6 nM T99347 C7C1WD 69085788 EC50 = 0.4 nM T99347 CHSO32 69086317 Ki = 10 nM T99347 C2QV3N 69092896 EC50 = 0.7 nM T99347 C9X2MF 69093210 Ki = 1.8 nM T99347 CLEO34 69093438 EC50 = 1.5 nM T99347 CXD2P5 69093459 EC50 = 14 nM T99347 CAO91L 69093544 EC50 = 4.8 nM T99347 C0JX3I 69093594 EC50 = 3.3 nM T99347 C8B1AL 69093815 EC50 = 10 nM T99347 C2J4PB 69093897 EC50 = 1.5 nM T99347 C67XGU 69093912 Ki = 1.4 nM T99347 C29WXD 69093963 EC50 = 1.2 nM T99347 CY80QV 69093997 EC50 = 0.2 nM T99347 CKS49I 69094308 EC50 = 9.4 nM T99347 CCE59I 69281818 Ki = 2.7 nM T99347 CZT05A 69929646 EC50 > 30000 nM T99347 CB0P8R 70654545 EC50 = 91 nM T99347 CKFN95 70681336 IC50 = 9300 nM T99347 CK7H9W 70681337 IC50 = 6000 nM T99347 CT91YG 70682455 EC50 = 390 nM T99347 CR1TI8 70682456 EC50 = 1100 nM T99347 C5ETU2 70682457 IC50 = 550 nM T99347 CF7LN2 70683431 IC50 = 4000 nM T99347 CNB8Z0 70684543 IC50 = 2100 nM T99347 CF7KR6 70686680 EC50 > 10000 nM T99347 C6E0DN 70686681 IC50 = 920 nM T99347 C4CK3B 70687684 IC50 = 9200 nM T99347 CS61RU 70687689 IC50 = 850 nM T99347 CRKV58 70688782 EC50 > 10000 nM T99347 C8XKB0 70688784 IC50 = 800 nM T99347 CY0C7Z 70690864 IC50 = 1600 nM T99347 CYI6J2 70690865 IC50 = 1100 nM T99347 C0RN7M 70693924 IC50 = 3900 nM T99347 C5TN8U 70695043 EC50 = 3200 nM T99347 CKAE71 70695044 EC50 = 2300 nM T99347 COPW78 70695204 EC50 = 460 nM T99347 CR7Y8S 70696165 IC50 = 8700 nM T99347 CH26LT 70957308 Ki = 23 nM T99347 CWT0H2 71449380 EC50 = 1400 nM T99347 CIYU65 71449381 IC50 = 2100 nM T99347 CQT2Y9 71449382 IC50 = 920 nM T99347 CVK81Z 71449383 IC50 = 390 nM T99347 CG5U1P 71449384 IC50 = 1800 nM T99347 C8B0HA 71449385 EC50 = 410 nM T99347 C6Z5LP 71449386 EC50 = 1000 nM T99347 COX4L6 71449387 EC50 = 1100 nM T99347 CQ6D4H 71449396 EC50 = 370 nM T99347 C8S7OD 71449397 EC50 = 865 nM T99347 CM5T4J 71449413 EC50 = 180 nM T99347 C51TWQ 71450775 EC50 > 10000 nM T99347 C0W7YK 71451180 EC50 = 6800 nM T99347 C90KNC 71451181 IC50 = 670 nM T99347 C4YA1Z 71451182 IC50 = 650 nM T99347 C29WHQ 71451183 EC50 = 500 nM T99347 CHI86F 71451184 IC50 = 1000 nM T99347 CCL8I2 71451192 EC50 = 540 nM T99347 C5Q6CJ 71451193 EC50 = 2200 nM T99347 CLAQ53 71451194 EC50 > 10000 nM T99347 CL2GX8 71451195 EC50 = 400 nM T99347 CMG8W3 71451196 EC50 = 72 nM T99347 C10TDI 71451334 IC50 = 31 nM T99347 CQV73C 71451335 IC50 = 65 nM T99347 CO48GV 71451554 IC50 = 3300 nM T99347 CY9QL3 71453007 IC50 = 670 nM T99347 C0G1XV 71453008 EC50 = 7100 nM T99347 CF9LN2 71453009 IC50 = 1300 nM T99347 CMKY72 71453020 EC50 = 680 nM T99347 C46RPK 71453021 EC50 = 200 nM T99347 CL61VS 71453022 EC50 = 1500 nM T99347 CSY6D5 71453023 EC50 = 74 nM T99347 CCQT65 71453150 IC50 = 11 nM T99347 C8X7PZ 71453151 IC50 = 670 nM T99347 CVUC16 71453394 IC50 = 176 nM T99347 CUP89A 71453395 IC50 = 4700 nM T99347 CJ2P1U 71454503 IC50 = 164 nM T99347 CX17UO 71454745 IC50 = 950 nM T99347 CX6HF9 71454746 IC50 = 1500 nM T99347 CJM13D 71454747 EC50 = 180 nM T99347 CVN6I5 71454754 EC50 = 47 nM T99347 CIM85E 71454886 IC50 = 4 nM T99347 CP7XR2 71454887 IC50 = 47 nM T99347 C8JT9X 71454888 IC50 = 540 nM T99347 C5ZQG4 71455089 IC50 = 1100 nM T99347 CQ4X8F 71456509 IC50 = 780 nM T99347 CW4N6U 71456510 IC50 = 170 nM T99347 CBTF29 71456511 IC50 = 130 nM T99347 C92HKN 71456512 IC50 = 1100 nM T99347 C97XUD 71456519 EC50 = 520 nM T99347 CJR4U0 71456520 IC50 = 1830 nM T99347 CQR9X1 71456521 IC50 = 990 nM T99347 CKAR73 71456522 EC50 > 10000 nM T99347 CMTW26 71456523 EC50 = 1900 nM T99347 CJU45V 71456662 IC50 = 240 nM T99347 CYI3G2 71456663 IC50 = 13 nM T99347 CA0K5X 71456664 IC50 = 300 nM T99347 CG5F7D 71456665 IC50 = 780 nM T99347 CQ3M4K 71458359 EC50 = 970 nM T99347 CD49FO 71458360 EC50 = 1000 nM T99347 C71VMQ 71458361 EC50 = 520 nM T99347 C8NOK9 71458362 EC50 = 1000 nM T99347 CWNJ29 71458371 EC50 = 2400 nM T99347 CN6YS1 71458372 IC50 = 920 nM T99347 CEU0N8 71458373 IC50 = 1400 nM T99347 C74ZPV 71458374 EC50 = 120 nM T99347 CFYU32 71458509 IC50 = 540 nM T99347 CQ8W7L 71459940 IC50 = 27 nM T99347 C6VG4H 71460197 IC50 = 4000 nM T99347 C7RBM6 71460198 EC50 = 2400 nM T99347 CG8WK0 71460199 EC50 = 1500 nM T99347 C0YH9L 71460214 IC50 = 3400 nM T99347 CKJ1H8 71460215 EC50 = 1200 nM T99347 CHE7N9 71460216 EC50 = 100 nM T99347 CE1B6D 71460217 EC50 = 98 nM T99347 CTJ8U7 71460353 IC50 = 3100 nM T99347 CLZO67 71460568 IC50 > 10000 nM T99347 C7KU6Q 71461917 IC50 = 1400 nM T99347 C9GTE2 71461918 EC50 = 2500 nM T99347 C71POQ 71461919 EC50 = 3200 nM T99347 CI51SO 71461920 EC50 = 950 nM T99347 C7JC3P 71461921 IC50 = 2500 nM T99347 CAG6P5 71461922 IC50 = 1900 nM T99347 CSR9F7 71461923 EC50 = 590 nM T99347 CET84J 71461924 IC50 = 890 nM T99347 CW1E6K 71461934 EC50 = 990 nM T99347 CI8G6W 71461935 IC50 = 1800 nM T99347 CWX12U 71462055 IC50 = 2700 nM T99347 CO6M5A 71462056 IC50 = 240 nM T99347 CNIW83 71479388 EC50 > 30000 nM T99347 CXP7O8 71479666 IC50 = 27.4 nM T99347 C04QUL 71521947 IC50 = 1.1 nM T99347 CO8D7T 71559536 IC50 = 27 nM T99347 CHGO45 71559676 IC50 > 10000 nM T99347 C4DSJ7 71560067 IC50 = 72 nM T99347 CEF36O 71560068 IC50 = 23 nM T99347 C0BDE3 71560069 Ki = 30 nM T99347 C75DUF 71560070 IC50 = 2910 nM T99347 CJR3D0 71560071 IC50 = 115 nM T99347 CO6WF0 71560072 IC50 > 10000 nM T99347 C9IW3Q 71560815 IC50 > 10000 nM T99347 C2SK9Z 71560816 IC50 > 10000 nM T99347 CJYN80 71560819 IC50 = 231 nM T99347 C8CNK9 71560943 IC50 > 10000 nM T99347 CKN8U1 71560944 IC50 > 10000 nM T99347 CKR5P0 71560945 IC50 = 314 nM T99347 CWZ0G7 71560946 IC50 = 62 nM T99347 CFU6C7 71560947 IC50 > 10000 nM T99347 C7BO9X 71560948 IC50 = 1510 nM T99347 CSP2A0 71561073 IC50 > 10000 nM T99347 CU4M9P 71561075 IC50 = 139 nM T99347 CJ5Z8R 71561198 IC50 = 671 nM T99347 CA1C3E 71561201 IC50 = 59 nM T99347 C95DZX 71561287 IC50 = 50 nM T99347 C6I7CG 71561313 IC50 = 9600 nM T99347 C6TER0 71561316 IC50 > 10000 nM T99347 CQOV51 71561317 IC50 = 5000 nM T99347 C6TEO9 71562957 IC50 = 430 nM T99347 C0NFT4 71563078 IC50 = 750 nM T99347 C26KRC 71573458 EC50 = 29 nM T99347 CBD9J0 71579830 IC50 = 4.4 nM T99347 CF4K1D 71579831 IC50 = 3.8 nM T99347 CN6AV0 71579832 IC50 = 4.7 nM T99347 CSMZ17 71579833 IC50 = 4.3 nM T99347 CE62ZG 71579924 IC50 = 3.7 nM T99347 CD61XW 71579925 IC50 = 5.3 nM T99347 C23GTO 71579926 IC50 = 2.3 nM T99347 CC4V3Q 71579927 IC50 = 5.3 nM T99347 CW4K5U 71579928 IC50 = 38 nM T99347 CHN16P 71579929 IC50 = 17 nM T99347 CQE4F0 71579930 IC50 = 645 nM T99347 CVE7X0 71580019 IC50 = 71 nM T99347 CL56RK 71580020 IC50 = 25 nM T99347 C4AWL6 71580021 IC50 = 92 nM T99347 C47GMF 71580022 IC50 = 1300 nM T99347 C4U0DH 71580120 IC50 = 911 nM T99347 C6K1RS 71580121 IC50 = 90.8 nM T99347 CUT53R 71580122 IC50 = 82.3 nM T99347 CS7DR1 71580123 IC50 = 16.4 nM T99347 C39XOZ 71580124 IC50 = 130 nM T99347 C83QIC 71580125 IC50 = 28 nM T99347 C8LM1R 71580126 IC50 = 195 nM T99347 C8EP1X 71580229 IC50 = 10.3 nM T99347 C9DHS8 71580230 IC50 = 184 nM T99347 CY1EL9 71580231 IC50 = 300.5 nM T99347 CHSD28 71580232 IC50 = 94.5 nM T99347 C3AG9H 71580233 IC50 = 56.3 nM T99347 CXQY46 71580234 IC50 = 41.6 nM T99347 CA92JC 71580235 IC50 = 7.1 nM T99347 CESN30 71580328 IC50 = 16.4 nM T99347 C6V7QA 71580329 IC50 = 2700 nM T99347 C1XGD9 71580331 IC50 = 5.8 nM T99347 C9OUN4 71580332 IC50 = 14.5 nM T99347 C7K2ML 71580333 IC50 = 147 nM T99347 CCD54K 71580334 IC50 = 46.2 nM T99347 CJA50E 71580442 IC50 = 17.1 nM T99347 C95SFQ 71580443 IC50 = 24.2 nM T99347 CL4QG9 71585302 EC50 = 53 nM T99347 C61EHT 71585509 EC50 = 73 nM T99347 C60EDU 71585613 EC50 = 272 nM T99347 C3XPL4 71585614 EC50 = 67 nM T99347 CP40YO 71585715 EC50 = 54 nM T99347 CXW32M 71585718 EC50 = 680 nM T99347 C1NY5O 71585719 EC50 = 38 nM T99347 CDL7M3 71585818 EC50 = 914 nM T99347 CMB08F 71585916 EC50 = 1527 nM T99347 C8CFV0 71586583 EC50 = 84 nM T99347 C78TOY 71586584 EC50 = 41 nM T99347 CMN0H6 71586585 EC50 = 858 nM T99347 CW46KS 71586682 EC50 = 76 nM T99347 C36CRV 71586683 EC50 = 53 nM T99347 C9Q7SY 71586684 EC50 = 97 nM T99347 C3R7ZH 71656663 EC50 = 224 nM T99347 C0SZM1 71656844 EC50 = 64 nM T99347 CS4J8H 71656937 EC50 = 431 nM T99347 CSQB24 71657122 EC50 = 769 nM T99347 C1AET0 71657125 EC50 = 61 nM T99347 C8L5KI 71657229 EC50 = 90 nM T99347 CQTW51 71712435 EC50 = 290 nM T99347 C5QE0A 71712436 EC50 = 2500 nM T99347 C73XAC 71712437 EC50 = 1500 nM T99347 CED28M 71712438 EC50 = 5200 nM T99347 CT4LI9 71712439 EC50 > 10000 nM T99347 CTD0V2 71712440 EC50 > 10000 nM T99347 CPF8H7 71712441 EC50 = 51 nM T99347 C6VXD0 71712576 EC50 = 2.5 nM T99347 C4VW2Y 71712577 IC50 = 23 nM T99347 CKV0D9 71712584 EC50 = 34 nM T99347 C9CVZ1 71712585 EC50 > 10000 nM T99347 CMJ89E 71712727 IC50 = 1200 nM T99347 C2K9QZ 71712728 IC50 = 72 nM T99347 CK6J0H 71712729 EC50 = 110 nM T99347 C6W1DJ 71712730 EC50 = 100 nM T99347 CI14UX 71712731 IC50 = 650 nM T99347 CT8Z1V 71712732 IC50 = 200 nM T99347 CH95RC 71712733 IC50 = 640 nM T99347 C5NP4T 71712734 IC50 = 400 nM T99347 C2HR6Y 71712876 EC50 > 10000 nM T99347 CB31DP 71712877 IC50 = 90 nM T99347 CX6B2J 71712878 IC50 = 38 nM T99347 CYNK39 71712879 IC50 = 290 nM T99347 CAB6X8 71712880 EC50 = 9.4 nM T99347 C9ZEQ6 71712881 EC50 = 3.9 nM T99347 CE3FH9 71712882 IC50 = 370 nM T99347 CY1K6E 71712883 EC50 = 81 nM T99347 CG95IA 71713016 EC50 = 17 nM T99347 C28KTU 71713017 EC50 = 85 nM T99347 CZ9E8U 71713018 EC50 = 18 nM T99347 CJ8RU6 71713019 EC50 = 2.5 nM T99347 C2C1ZQ 71713020 EC50 = 150 nM T99347 CU16TP 71713021 EC50 = 640 nM T99347 C0H9YL 71713022 EC50 = 19 nM T99347 CMC0Y3 71713169 EC50 = 130 nM T99347 CJWY24 71713170 EC50 = 790 nM T99347 C52VRK 71713171 EC50 = 167 nM T99347 C0CT4V 71713172 EC50 = 70 nM T99347 CNL51W 71713173 EC50 = 190 nM T99347 CE4SO9 71713174 EC50 = 100 nM T99347 C2RU3P 71713175 EC50 = 290 nM T99347 C64XUS 71713321 EC50 = 320 nM T99347 CFC30V 71713322 EC50 = 470 nM T99347 CE5J0B 71713324 EC50 = 1200 nM T99347 C1FN2E 71713325 EC50 = 99 nM T99347 CL7T3R 71713326 EC50 = 8.7 nM T99347 CBYD26 71713327 EC50 = 30 nM T99347 CA19EY 71713464 EC50 = 71 nM T99347 C8IQX6 71713465 EC50 = 11 nM T99347 CN2W7X 71713466 EC50 = 29 nM T99347 CX13NZ 71713467 EC50 = 160 nM T99347 CAR84Y 71713468 EC50 = 220 nM T99347 CSLX54 71713469 EC50 = 1600 nM T99347 C0K7EV 71713470 IC50 = 11 nM T99347 CXL0S3 71713607 IC50 = 140 nM T99347 C2MTL0 71713608 IC50 = 5.7 nM T99347 CP2K5R 71713609 IC50 = 34 nM T99347 CM5G7Y 71713610 IC50 = 36 nM T99347 CQF67U 71713611 IC50 = 480 nM T99347 CNK4L7 71713612 EC50 = 150 nM T99347 CTZ6L2 71713613 IC50 = 780 nM T99347 CQMH24 71713761 EC50 = 250 nM T99347 CK6N5Z 71713762 IC50 = 13 nM T99347 C3FK4C 71713763 EC50 = 75 nM T99347 CG3ZS0 71713764 EC50 = 72 nM T99347 CH23SQ 71713765 EC50 = 74 nM T99347 CGUK74 71713766 EC50 = 9.8 nM T99347 C1D0HO 71713767 EC50 = 53 nM T99347 CZM41U 71713920 EC50 = 26 nM T99347 CD5EO9 71713921 EC50 > 10000 nM T99347 CI3N1E 71716502 IC50 = 468 nM T99347 CW9N3L 71716503 IC50 = 228 nM T99347 CAS1F0 71717012 IC50 = 47 nM T99347 CL48YV 71717107 IC50 > 10000 nM T99347 C0GF7R 71717108 IC50 = 789 nM T99347 CZY7D1 71717109 IC50 > 10000 nM T99347 CF03TE 71717110 IC50 = 857 nM T99347 C25HCQ 71717116 IC50 = 139 nM T99347 CZTX70 71717117 IC50 = 88.3 nM T99347 CXS25P 71717644 IC50 = 36 nM T99347 C4AJ8X 71717729 IC50 = 266 nM T99347 C56XPS 71717730 IC50 = 7840 nM T99347 C1LIE9 71717735 IC50 = 77 nM T99347 CC9B6X 71717783 IC50 > 1000 nM T99347 C2WU9T 71717784 IC50 > 1000 nM T99347 CMUZ70 71718339 IC50 = 1000 nM T99347 C75TFV 71718340 IC50 = 593 nM T99347 COCW75 71718341 IC50 = 300 nM T99347 CKXM23 71718937 IC50 = 531 nM T99347 CLC0S8 71718938 IC50 = 290 nM T99347 C2YOD7 71718942 IC50 = 62 nM T99347 CV34BP 71718943 IC50 = 27 nM T99347 CC2VP4 71719552 IC50 = 175 nM T99347 C60QUO 71719558 IC50 = 40.4 nM T99347 CM10TY 71720053 IC50 = 35 nM T99347 C9G3LC 71720146 IC50 = 1370 nM T99347 CXJ3P6 71720147 IC50 = 425 nM T99347 CLUP87 71720148 IC50 = 612 nM T99347 C06IWM 71720149 IC50 = 3400 nM T99347 C9RUK0 71720153 IC50 = 12 nM T99347 CB1LC6 71720791 IC50 = 86 nM T99347 CW7QS2 71720792 IC50 = 194 nM T99347 CS1P4T 71720793 IC50 = 473 nM T99347 C49YUD 71720794 IC50 = 1150 nM T99347 CQH0Z4 71720798 IC50 = 173 nM T99347 C19ALP 71720843 IC50 = 27 nM T99347 C7R5MI 71720844 IC50 = 95 nM T99347 C62KPZ 71743756 IC50 > 100000 nM T99347 CTB63F 71812961 IC50 = 11000 nM T99347 C1JRI7 71812962 IC50 > 100000 nM T99347 CQ1N6P 71812963 EC50 = 694 nM T99347 CC20YE 71813137 IC50 > 100000 nM T99347 C6EC3O 72163432 IC50 = 3360 nM T99347 CNF81W 72163837 IC50 > 10000 nM T99347 CZ0G2X 72165213 Ki = 0.9 nM T99347 CWJH59 72545303 IC50 = 298 nM T99347 C6LX1H 72545304 IC50 = 61.3 nM T99347 CO80FA 72545305 IC50 = 2190 nM T99347 CY7DP1 72545306 IC50 = 46.6 nM T99347 CMG27Z 72545550 IC50 = 187 nM T99347 C7QYG8 72545551 IC50 = 72.2 nM T99347 CEA67F 72545553 IC50 = 818 nM T99347 C2QEZ0 72545554 IC50 > 100000 nM T99347 CI0D5R 72545802 IC50 = 543 nM T99347 CD8JI0 72545803 IC50 = 308 nM T99347 CE82JD 72545804 IC50 = 47.8 nM T99347 CGVS93 72545805 IC50 = 132 nM T99347 CI38QZ 72545807 IC50 = 210 nM T99347 CCA7G8 72546040 IC50 = 168 nM T99347 C3KG1F 72546042 IC50 = 575 nM T99347 C8V6GX 72546044 IC50 = 170 nM T99347 COB7Z8 72546271 IC50 = 64.8 nM T99347 CZJ5P9 72546272 IC50 = 137 nM T99347 CF8R5E 72546273 IC50 = 1020 nM T99347 C6HA8S 72546277 IC50 = 3350 nM T99347 CSY2K7 72546509 IC50 = 36.5 nM T99347 C4PTL6 72546510 IC50 = 930 nM T99347 CXZ72O 72546514 IC50 = 227 nM T99347 CT0R1O 72546751 IC50 = 306 nM T99347 C4HF5O 72546752 IC50 = 813 nM T99347 CJ4S3D 72546753 IC50 = 340 nM T99347 CCBI73 72546754 IC50 = 86.3 nM T99347 C41XHL 72546755 IC50 = 76.3 nM T99347 CXW8R2 72714783 EC50 = 158.49 nM T99347 C96CJO 73346313 EC50 = 717 nM T99347 C28DPN 73346314 EC50 = 40 nM T99347 CK4DH9 73347520 EC50 = 18 nM T99347 C9OUV5 73349072 IC50 > 100000 nM T99347 CMDO68 73352407 EC50 = 90 nM T99347 C6J9BZ 73356665 IC50 > 100000 nM T99347 CBS3X1 73603977 IC50 = 90 nM T99347 CZ3TB5 74221949 IC50 = 54 nM T99347 C7L5NU 74221951 IC50 = 58 nM T99347 CW9N8T 74222036 IC50 = 63 nM T99347 CPR6D0 76309825 IC50 = 28.4 nM T99347 C95SLK 76310873 Ki = 26 nM T99347 C4URX9 76310874 Ki = 7.8 nM T99347 C7LPF6 76318078 Ki = 899 nM T99347 C3Z2CN 76320761 IC50 = 180 nM T99347 CQ5ZT1 76321784 Ki = 8.1 nM T99347 COF43E 76321785 Ki = 54.6 nM T99347 CGV1R4 76321786 Ki = 6.6 nM T99347 C1D0YN 76324428 IC50 = 1010 nM T99347 CZ63YO 76325409 Ki = 5 nM T99347 C5KTM1 76325410 Ki = 1.3 nM T99347 C5BY7D 76325411 Ki = 42 nM T99347 CM2N7X 76328023 IC50 = 103 nM T99347 C94QVX 76328949 Ki = 6.2 nM T99347 C6MC3A 76328950 Ki = 2.3 nM T99347 CZ0XA2 76328951 Ki = 11 nM T99347 CQR84K 76328952 Ki = 2.8 nM T99347 CR2F5W 76328953 Ki = 7 nM T99347 CL92TU 76328954 Ki = 10 nM T99347 CWJA51 76328955 Ki = 4.85 nM T99347 C7SE2H 76331633 IC50 = 8600 nM T99347 CH2J7R 76331684 IC50 = 85 nM T99347 CTE1J7 76332628 Ki = 58 nM T99347 C80MQG 76332629 Ki = 114 nM T99347 CXK8Y7 76335252 IC50 = 189 nM T99347 CM69HE 76336232 Ki = 11 nM T99347 CI2P5S 76336233 Ki = 6.5 nM T99347 CHP5I0 76570032 Ki = 276 nM T99347 CIZ52U 86280685 Ki = 0.5012 nM T99347 CG1RU5 86627336 Ki = 0.3 nM T99347 CQ45XR 86763358 Ki = 0.5012 nM T99347 CT6D2J 87549991 Ki = 0.3 nM T99347 CSRU90 87550393 Ki = 2.7 nM T99347 CE0MR2 87550659 Ki = 0.5 nM T99347 CTJ6D7 87550873 Ki = 0.5 nM T99347 C0C1TK 87551058 Ki = 83 nM T99347 CWE0N6 90646585 Ki = 1.259 nM T99347 COC4K8 90646677 Ki = 3.981 nM T99347 C9J7DF 90646679 Ki = 2.512 nM T99347 CBDQ30 90646779 Ki = 1.585 nM T99347 CIC3X1 91668258 IC50 = 0.3981 nM T99347 C0KVB7 99941396 Ki = 6.1 nM T99347 CT6F1D 117820994 IC50 = 2.512 nM T99347 CX91IL 117821459 Ki = 10 nM T99347 CD0Z9U 117821593 IC50 = 0.631 nM T99347 C32FYH 117824339 Ki = 1.585 nM T99347 C9F4ZD 118008435 Ki = 17 nM T99347 CLO18J 118008580 EC50 > 1600 nM T99347 CZ1V0Y 118008603 Ki = 30 nM T99347 CUGO65 118008663 EC50 = 250 nM T99347 CHZ0U1 118008796 Ki = 1667 nM T99347 C0YMS9 118008803 Ki = 36 nM T99347 CCQ42L 118008809 Ki = 580 nM T99347 CQ68CV 118008894 EC50 = 90 nM T99347 CW8ID5 118019330 Ki = 47 nM T99347 COG2R3 118019339 EC50 = 77 nM T99347 C9T5VI 118019340 EC50 = 8 nM T99347 C7GB0U 118019347 EC50 = 31 nM T99347 CRQ6O1 118019350 Ki = 259 nM T99347 CW3L7K 118019351 Ki = 67 nM T99347 CO6PY8 118019352 Ki = 47 nM T99347 CL1S6H 118019353 Ki = 13 nM T99347 C2C5EH 118019356 Ki = 108 nM T99347 C35NPI 118019357 EC50 = 18 nM T99347 C5KW2Z 118019359 EC50 = 13 nM T99347 CU8BG5 118019360 EC50 = 35 nM T99347 CN7J0H 118019361 Ki = 59 nM T99347 CD5P0X 118204277 IC50 = 31.2 nM T99347 C6B1FH 118204278 IC50 = 27.8 nM T99347 C3EUC0 118204279 IC50 = 10 nM T99347 CCGE86 118204291 IC50 = 8.2 nM T99347 CW57PO 118204292 IC50 = 15.4 nM T99347 C9A2XY 118204293 IC50 = 9.3 nM T99347 CE86VG 118204300 IC50 = 182 nM T99347 CZB5Y4 118204305 IC50 = 23.3 nM T99347 CI7A1V 118204306 IC50 = 30.9 nM T99347 CJV15O 118204307 IC50 = 16.6 nM T99347 CQ4K9T 118204308 IC50 = 37.8 nM T99347 CLI31P 118204320 IC50 = 42.2 nM T99347 CSY4J8 118204338 IC50 = 13.3 nM T99347 CB1D9J 118204339 IC50 = 2.4 nM T99347 C2OLR1 118204347 IC50 = 7.5 nM T99347 CKM2U6 118204375 IC50 = 978 nM T99347 CXQ4R7 118204378 IC50 = 9.7 nM T99347 CL4AK7 118204489 IC50 = 12.8 nM T99347 C7SYF3 118204617 IC50 = 30.9 nM T99347 CRQ5W1 118609053 IC50 = 388 nM T99347 C9WOZ2 118612903 IC50 = 2330 nM T99347 CMW3K0 118612909 IC50 = 725 nM T99347 C38GYS 118612925 IC50 = 31 nM T99347 CM4HO1 118612935 IC50 = 228 nM T99347 CNG98M 118612937 IC50 = 51 nM T99347 CJQ0T2 118612938 IC50 = 899 nM T99347 C08NIG 118612946 IC50 = 43 nM T99347 C3EOF6 118612948 IC50 = 66 nM T99347 C62KBZ 118612952 IC50 = 140 nM T99347 C92SOF 118612955 IC50 = 902 nM T99347 CA83HB 118612958 IC50 = 273 nM T99347 CI0N6C 118612960 IC50 = 210 nM T99347 CQ5WS4 118612962 IC50 = 700 nM T99347 CSMT69 118612971 IC50 = 145 nM T99347 C1UQ7W 118612974 IC50 = 504 nM T99347 CM19WK 118612993 IC50 = 200 nM T99347 C2J3MI 118613016 IC50 = 182 nM T99347 CLCA57 118613025 IC50 = 180 nM T99347 CFW8M4 118613034 IC50 = 1420 nM T99347 CX5C3F 118613043 IC50 = 1960 nM T99347 CD8GA6 118613045 IC50 = 5200 nM T99347 C6R1CI 118613047 IC50 = 3350 nM T99347 C4D0WV 118613049 IC50 = 392 nM T99347 C9SDJ7 118613050 IC50 = 2100 nM T99347 CT41HO 118613057 IC50 = 1560 nM T99347 C8G0HR 118613058 IC50 = 497 nM T99347 CFT3M9 118613060 IC50 = 646 nM T99347 CX6Q3U 118613066 IC50 = 149 nM T99347 C1IBC0 118613068 IC50 = 175 nM T99347 C6AG2L 118613071 IC50 = 4470 nM T99347 CGY3J6 118613074 IC50 = 932 nM T99347 C9R7XI 118613075 IC50 = 399 nM T99347 C5H1BQ 118613081 IC50 = 58 nM T99347 CLO16W 118613086 IC50 = 1050 nM T99347 CBEX87 118613088 IC50 = 224 nM T99347 CKRM87 118613091 IC50 = 446 nM T99347 C5N3IC 118613130 IC50 = 182 nM T99347 C2NRI0 118613132 IC50 = 3660 nM T99347 CL5R7Z 118613136 IC50 = 684 nM T99347 CVW15G 118613138 IC50 = 1290 nM T99347 CZTJ92 118613141 IC50 = 194 nM T99347 CBC0M8 118613143 IC50 = 2480 nM T99347 C89JZV 118613144 IC50 = 134 nM T99347 CK6TB7 118613145 IC50 = 38 nM T99347 C0OWB4 118613147 IC50 = 81 nM T99347 C6NSY1 118613150 IC50 = 392 nM T99347 C5AVX2 118613153 IC50 = 4300 nM T99347 C2ZH4X 118613167 IC50 = 657 nM T99347 CW2N5S 118613172 IC50 = 107 nM T99347 CWX75R 118613174 IC50 = 23 nM T99347 CP7W9O 118613176 IC50 = 28 nM T99347 CHV9R0 118613253 IC50 = 145 nM T99347 C6RUO7 118613255 IC50 = 1030 nM T99347 CM02XS 118613397 IC50 = 77 nM T99347 CS4R3B 118707826 IC50 = 85 nM T99347 CON8L2 118732212 Ki = 1770 nM T99347 CZ48DA 118732213 IC50 = 26 nM T99347 C0JEU5 118732214 Ki = 2840 nM T99347 CV5RN4 118732215 IC50 = 124 nM T99347 CH69NQ 118732216 Ki = 255 nM T99347 C86VAW 118732217 IC50 = 9 nM T99347 CS3P1A 118732218 IC50 = 11 nM T99347 CS26JL 118732219 IC50 = 13 nM T99347 C70UKD 118732220 IC50 = 100 nM T99347 C8NSP0 118732221 IC50 = 141 nM T99347 C8CP2R 118732222 IC50 = 295 nM T99347 CDA98H 118735955 IC50 = 4830 nM T99347 C5P0XW 118735974 IC50 = 1430 nM T99347 CPGY12 118735978 IC50 = 4730 nM T99347 C7BL9C 122183731 Ki = 0.4 nM T99347 CWME54 122183732 IC50 = 42 nM T99347 CD78GJ 122183733 Ki > 10000 nM T99347 CFM0Y3 122183734 Ki > 10000 nM T99347 CQ38OP 122183735 Ki > 10000 nM T99347 CE87FS 122183736 Ki > 10000 nM T99347 CKRW37 122183737 Ki = 283.1 nM T99347 C7L6GM 122183738 Ki = 0.3 nM T99347 C7GL0N 122183739 Ki = 41.8 nM T99347 CKWS56 122184229 IC50 = 71.4 nM T99347 C95CYS 122184231 IC50 = 60 nM T99347 CDN19B 122184232 IC50 = 43.9 nM T99347 C20NUE 122184233 IC50 = 584 nM T99347 CEHV90 122185251 IC50 > 1000 nM T99347 CV0N8K 122185252 IC50 = 1055 nM T99347 C5ZJ3K 122185253 IC50 > 1000 nM T99347 C4KJ8V 122185254 IC50 = 8.8 nM T99347 CRJ12E 122185255 IC50 = 55.5 nM T99347 CXI5O4 122185256 IC50 = 55.9 nM T99347 CV9LA0 122185325 Ki = 63.1 nM T99347 CPB38M 122185326 Ki = 251.19 nM T99347 CO38ZV 122185327 Ki = 794.33 nM T99347 C17BEL 122185328 Ki = 7943.28 nM T99347 C75ZOS 122185329 Ki > 63095.73 nM T99347 CW9A6M 122185330 Ki > 63095.73 nM T99347 CUS9Q5 122185331 Ki = 25.12 nM T99347 CU1BC8 122185332 Ki = 19.95 nM T99347 C24HOQ 122185333 Ki = 19.95 nM T99347 C71PLQ 122185334 Ki = 5.012 nM T99347 CU0XJ3 122186361 EC50 > 10000 nM T99347 CO9P2G 122186362 EC50 = 323.59 nM T99347 C7W5XH 122186363 EC50 = 750 nM T99347 CF1C0Q 122186364 EC50 = 510 nM T99347 C1L4AJ 122186365 EC50 = 520 nM T99347 CUFP39 122186366 EC50 = 170 nM T99347 CUC13P 122187795 IC50 > 30000 nM T99347 CCP5U2 122195692 EC50 = 360 nM T99347 C67JPK 122195693 EC50 = 331.13 nM T99347 CCF57J 122195694 EC50 = 1698.24 nM T99347 C5R4WI 122195695 EC50 = 882 nM T99347 CZ5UA3 122195696 EC50 = 524.81 nM T99347 C68CVY 122195697 EC50 = 1220 nM T99347 C49MNU 122195698 EC50 = 1737.8 nM T99347 CS9O3F 122195699 EC50 = 371.54 nM T99347 C4SGA0 122195700 EC50 = 610 nM T99347 CRX6Z1 122195701 EC50 = 1122.02 nM T99347 C1TAL0 122195702 EC50 = 588.84 nM T99347 CH2G7X 122195703 EC50 = 596 nM T99347 CS5K7P 122195704 EC50 = 389.05 nM T99347 C6D5IJ 122195705 EC50 > 10000 nM T99347 CA98LD 122195706 EC50 > 10000 nM T99347 CV2G6T 122195707 EC50 > 31622.78 nM T99347 C76MSF 122195708 EC50 = 2754.23 nM T99347 C93LJZ 122195709 EC50 = 257 nM T99347 C7S8CE 122195710 EC50 = 2344.23 nM T99347 CK9L6F 122195711 EC50 = 239.88 nM T99347 CT85AD 122195712 EC50 > 10000 nM T99347 C0PTS3 122195713 EC50 = 1258.93 nM T99347 C7T4ZC 122195714 EC50 > 10000 nM T99347 CV0G8T 122195715 EC50 > 31622.78 nM T99347 C0P9AY 122195716 EC50 > 31622.78 nM T99347 CT12WE 122195717 EC50 = 3890.45 nM T99347 CS7GH5 122195718 EC50 > 31622.78 nM T99347 CAJ3F7 122195719 EC50 > 31622.78 nM T99347 CJ64HQ 122195720 EC50 > 10000 nM T99347 C4DZ5R 122195721 EC50 = 700 nM T99347 C1V3DP 122195722 EC50 > 31622.78 nM T99347 CBW28T 122195723 EC50 > 31622.78 nM T99347 C4V0AB 122195724 EC50 > 10000 nM T99347 CR86EO 122195725 EC50 = 724.44 nM T99347 CEQS83 122195726 EC50 = 794 nM T99347 COLG41 122195727 EC50 = 5370 nM T99347 CE7P9D 122195728 EC50 = 3400 nM T99347 CC4L6G 122195898 EC50 = 780 nM T99347 CAE90O 122195899 EC50 = 888 nM T99347 C4DG3Y 122195900 EC50 = 1345 nM T99347 C2HW9X 122195901 EC50 = 3236 nM T99347 CYW2D4 122459067 EC50 = 237 nM T99347 CG9H8V 122459068 EC50 = 300 nM T99347 CH2AO4 122539788 IC50 > 30000 nM T99347 CB2ZK5 127026165 EC50 > 10000 nM T99347 C7J5VX 127026166 EC50 > 10000 nM T99347 C9XU8I 127026167 EC50 > 10000 nM T99347 CA42BO 127027101 EC50 > 10000 nM T99347 C09CHL 127027102 EC50 > 10000 nM T99347 CGI3P5 127034893 EC50 = 31.62 nM T99347 CGY60A 127034894 EC50 = 15.85 nM T99347 CCX0U4 127034895 EC50 = 1584.89 nM T99347 C2A6XR 127034896 EC50 = 1258.93 nM T99347 CWDX89 127034897 EC50 = 199.53 nM T99347 C4NQ6X 127034898 EC50 = 19.95 nM T99347 C4GIU2 127035061 EC50 = 1000 nM T99347 CQ87IO 127035182 EC50 > 25118.86 nM T99347 CQ6OI4 127035365 EC50 = 79.43 nM T99347 CM21DZ 127035366 EC50 = 5.012 nM T99347 CV2XI1 127035885 EC50 = 1000 nM T99347 C2KC9W 127035890 EC50 = 50.12 nM T99347 C9TYJ6 127036276 EC50 = 10 nM T99347 CX3N1Y 127036699 EC50 = 15.85 nM T99347 C3W1NG 127036700 EC50 = 3981.07 nM T99347 C8SM0I 127036904 EC50 = 398.11 nM T99347 COG5K7 127036905 EC50 = 398.11 nM T99347 CE65UK 127036906 EC50 = 5.012 nM T99347 C2TRB4 127037297 EC50 = 31.62 nM T99347 CI2Y0S 127037639 EC50 = 3162.28 nM T99347 C21KEJ 127038586 EC50 > 30000 nM T99347 C1RY8E 127038766 IC50 = 274 nM T99347 C9I2BV 127039660 EC50 = 87.1 nM T99347 CR31FQ 127042313 IC50 = 159 nM T99347 CPZ70S 127052897 EC50 > 30000 nM T99347 C7FSD5 129012190 EC50 = 47 nM T99347 C38BRY 131801162 EC50 > 10000 nM T99347 CFC05Q 131954513 EC50 > 10000000 nM T99347 CC9IK3 132530619 EC50 = 120 nM T99347 CD1A2K 132530622 EC50 = 53 nM T99347 CAW69C 132530624 EC50 = 530 nM T99347 CO7I2Z 132530625 EC50 = 30 nM T99347 CIVX01 134132348 EC50 = 1300 nM T99347 C8ID6O 134132797 EC50 = 1400 nM T99347 CPX0E5 134132914 EC50 = 220 nM T99347 CAU26V 134135881 EC50 = 51 nM T99347 CL89ND 134136288 EC50 = 45 nM T99347 C5MQS1 134136925 EC50 = 49 nM T99347 CA38IJ 134137269 EC50 = 110 nM T99347 CXM56Y 134137686 EC50 = 31 nM T99347 CT0SI8 134139139 EC50 = 2360 nM T99347 CZ14MP 134139501 EC50 = 83 nM T99347 CQ7Y0F 134141244 EC50 = 190 nM T99347 CJT27E 134141319 EC50 = 150 nM T99347 CWS62X 134144704 EC50 > 3000 nM T99347 CU7KJ1 134144969 EC50 = 69 nM T99347 CJL15C 134147277 EC50 = 240 nM T99347 C8DVS1 134148604 EC50 = 140 nM T99347 C8RG2K 134151206 EC50 = 71 nM T99347 CL7C5I 134151933 EC50 = 21 nM T99347 C48BWR 134157129 EC50 = 330 nM T99347 C5YRP0 135659063 Ki = 6.761 nM T99347 C9NL5B 136058486 IC50 = 96 nM T99347 CKD3Z6 136058487 IC50 = 100 nM T99347 CYXS60 136082888 IC50 = 50 nM T99347 CL2NW4 136244237 IC50 > 12500 nM T99347 C63RDU 136254202 IC50 = 2400 nM T99347 CK4PX6 136254203 IC50 = 870 nM T99347 CSA4H8 136254204 IC50 = 1200 nM T99347 C3FPW2 136254205 IC50 = 250 nM T99347 CHU3Z5 136254206 IC50 = 570 nM T99347 C3EGM5 137321168 IC50 > 10000 nM T99347 CMT58F 137633212 Ki = 1 nM T99347 CE3H7S 137634667 IC50 = 237 nM T99347 C1WLT3 137634749 Ki = 194 nM T99347 CNU0H2 137635120 Ki = 3.8 nM T99347 CUC83P 137636158 IC50 = 157 nM T99347 CN7WD9 137638572 Ki = 24.1 nM T99347 CV6QR7 137639779 Ki = 98 nM T99347 CQ5LO9 137644273 Ki = 3.3 nM T99347 C16IRJ 137644674 Ki = 7 nM T99347 C0U3PG 137645039 Ki = 10 nM T99347 CS6N3B 137645412 IC50 = 403 nM T99347 C0AD8O 137645894 Ki = 5.5 nM T99347 C8Q0GD 137646682 IC50 = 177 nM T99347 C6JXQ1 137650553 Ki = 4 nM T99347 C8MKP2 137650972 Ki = 16 nM T99347 C0NSQ2 137653178 Ki = 1.5 nM T99347 C0Z3ME 137655893 Ki = 3 nM T99347 CZC0S4 137655976 Ki = 31 nM T99347 C57FIL 137658291 Ki = 27 nM T99347 CEJ7Y9 137658590 IC50 = 174 nM T99347 CV1ZN8 137659056 Ki = 15 nM T99347 C93RAP 137661535 Ki = 10 nM T99347 CX81OE 137661622 Ki = 30.9 nM T99347 CA1VK5 140268006 IC50 = 244 nM T99347 CFR6U7 140268009 IC50 = 150 nM T99347 CQR1B4 140268012 IC50 = 150 nM T99347 CO3BA8 140268020 IC50 = 164 nM T99347 C1C2PD 145949977 Ki > 10000 nM T99347 C5Z1LS 145952217 Ki > 10000 nM T99347 CSA16D 145952244 Ki > 10000 nM T99347 CD8I3S 145953412 Ki = 3077 nM T99347 C1AMD5 145955192 Ki = 1883 nM T99347 CGM3L7 145957163 Ki > 10000 nM T99347 C3W0QX 145957790 Ki > 10000 nM T99347 C7GH8Z 145960052 Ki > 10000 nM T99347 CNE72W 145982756 IC50 = 1600 nM T99347 CE2HG1 145983104 IC50 = 110 nM T99347 CWI9T1 145983268 IC50 = 240 nM T99347 CO84BZ 145983763 IC50 = 310 nM T99347 C1RI8D 145984337 IC50 = 1200 nM T99347 CXTG03 145984446 IC50 = 900 nM T99347 CXU69G 145984484 IC50 = 170 nM T99347 CC5KA9 145985295 IC50 = 320 nM T99347 CI93CR 145985513 IC50 = 2600 nM T99347 C8F4JV 145985945 IC50 = 450 nM T99347 C3IL9H 155511336 IC50 > 30000 nM T99347 CN25JM 155511343 IC50 > 10000 nM T99347 CMR0I8 155511389 IC50 = 1293 nM T99347 CZD2M7 155513245 IC50 = 257 nM T99347 C17RIB 155513592 Ki = 0.98 nM T99347 C5KD7U 155513648 IC50 = 270 nM T99347 C9HG0U 155515457 Ki = 5.8 nM T99347 CQ52LM 155518361 Ki = 2 nM T99347 C18EFY 155518933 EC50 = 630.96 nM T99347 CH5PY3 155519291 IC50 = 127 nM T99347 C1U3CL 155520250 Ki = 3.9 nM T99347 CD39ZJ 155520820 IC50 = 120 nM T99347 CXC63W 155522099 IC50 = 389 nM T99347 C0BH3X 155523654 IC50 = 9469 nM T99347 C4YNK7 155524301 IC50 = 2477 nM T99347 CFM45O 155524794 Ki = 2.9 nM T99347 C0HA5P 155527447 IC50 = 176 nM T99347 CW10CQ 155527469 IC50 = 7200 nM T99347 C75NEB 155529408 IC50 = 694 nM T99347 CK5X2E 155530190 Ki = 8.6 nM T99347 CQD26H 155530468 Ki = 38.3 nM T99347 CDE89R 155531760 IC50 = 383 nM T99347 CWJ18H 155534147 IC50 = 451 nM T99347 CTH8B9 155535743 Ki = 2.6 nM T99347 CY97DN 155535886 Ki = 0.7 nM T99347 CIM71P 155536796 IC50 = 395 nM T99347 CM1BX0 155537411 Ki = 4 nM T99347 CYXE53 155538270 IC50 > 10000 nM T99347 C3LXB4 155540022 IC50 = 2040 nM T99347 C2TVN9 155545208 IC50 = 112 nM T99347 CZ7NH0 155545491 IC50 > 30000 nM T99347 CH08FR 155547194 IC50 = 197 nM T99347 C08YOZ 155549638 Ki = 2.5 nM T99347 CEN69O 155549742 IC50 = 482 nM T99347 C2X8VM 155549812 IC50 = 201 nM T99347 CD4PW8 155550069 Ki = 243 nM T99347 CCA4D9 155551000 IC50 = 103 nM T99347 CGDS14 155551776 IC50 = 6.4 nM T99347 C7JH8N 155552861 Ki = 4 nM T99347 CE87BL 155554359 IC50 > 10000 nM T99347 C3Z4QS 155554969 Ki = 3.6 nM T99347 C8Q2FG 155555556 Ki = 3.5 nM T99347 C9H1VK 155556442 IC50 = 235 nM T99347 CGZM78 155557326 Ki > 1000 nM T99347 C5QLH0 155558779 IC50 = 568 nM T99347 CHP06O 155566645 IC50 > 10000 nM T99347 C2TNU1 155568511 IC50 = 477 nM T99347 CAFQ03 71458026 IC50 = 10 nM T99347 D00HIH 53252525 EC50 = 52 nM T99347 D00JUO 53380924 Ki = 12 nM T99347 D00NCL 46836562 EC50 > 10000 nM T99347 D01AJZ 11242036 IC50 = 1150 nM T99347 D01ALS 11535796 IC50 = 475 nM T99347 D01DPN 11572145 IC50 = 1243 nM T99347 D01ECL 11063448 IC50 = 53 nM T99347 D01ERW 11175501 IC50 = 5400 nM T99347 D01EVA 6278000 Ki > 100000 nM T99347 D01SYO 11095641 IC50 = 122 nM T99347 D01UUH 11564671 IC50 = 789 nM T99347 D01YEN 1233 Ki = 17000 nM T99347 D02BFK 11701423 IC50 = 129 nM T99347 D02DOP 10236192 IC50 = 3600 nM T99347 D02KHF 44403640 IC50 = 106 nM T99347 D02NMN 23634102 IC50 > 3000 nM T99347 D02NNU 16659803 IC50 > 1000 nM T99347 D02XFR 899301 IC50 = 15000 nM T99347 D03CCP 11550377 IC50 = 2920 nM T99347 D03LCM 44412923 IC50 = 12700 nM T99347 D03NFW 11772954 IC50 > 3000 nM T99347 D03NIO 11600877 IC50 = 946 nM T99347 D03NYF 44392959 IC50 = 22 nM T99347 D03OLR 71559428 IC50 = 20 nM T99347 D03PGL 46911068 EC50 > 10000 nM T99347 D03QRG 16735840 IC50 = 2.3 nM T99347 D04BES 11379837 IC50 = 5 nM T99347 D04DKM 104766 Ki = 15000 nM T99347 D04ILS 44409846 Ki = 5 nM T99347 D04JKL 2071 Ki > 1000000 nM T99347 D04MVR 11530404 IC50 = 442 nM T99347 D04PBZ 11564861 IC50 = 49 nM T99347 D04RVW 44392990 IC50 = 0.5 nM T99347 D04RYE 46866192 IC50 > 3000 nM T99347 D05AJJ 51346799 EC50 = 44.3 nM T99347 D05DCW 46866191 IC50 > 3000 nM T99347 D05FCO 12811064 IC50 = 3.1 nM T99347 D05FEO 72551298 EC50 = 33 nM T99347 D05KSC 11515548 IC50 = 4040 nM T99347 D05TFE 5218788 IC50 = 370 nM T99347 D05XNS 44412879 IC50 = 18300 nM T99347 D06DUE 40539 Ki = 55 nM T99347 D06KVX 11665793 IC50 = 36.3 nM T99347 D06PAK 10058694 Ki > 100000 nM T99347 D06PTC 44416004 IC50 = 258 nM T99347 D06TYA 16659967 IC50 > 1000 nM T99347 D06YKH 11536470 IC50 = 526 nM T99347 D06ZBT 11701860 IC50 = 60 nM T99347 D07FVZ 9931205 EC50 = 150 nM T99347 D07FXC 11299421 IC50 = 1540 nM T99347 D07GRG 10197984 Ki > 100000 nM T99347 D07JLC 3410100 IC50 = 10800 nM T99347 D07QJQ 10921526 IC50 = 4 nM T99347 D07RRA 11608117 IC50 = 1830 nM T99347 D08ADI 44409820 Ki = 58 nM T99347 D08FDI 9813637 IC50 = 270 nM T99347 D08FEV 11586785 IC50 = 1000 nM T99347 D08NQW 3645780 EC50 = 750000 nM T99347 D08PDF 4074142 IC50 = 486 nM T99347 D08SSG 11615445 IC50 = 698 nM T99347 D09AQK 4545574 Ki > 500000 nM T99347 D09GMG 585532 IC50 = 46000 nM T99347 D09LDM 11579392 IC50 = 2 nM T99347 D09QUN 58368068 EC50 = 70 nM T99347 D09UBS 10428048 Ki > 100000 nM T99347 D0AG1Q 11206949 IC50 = 28 nM T99347 D0B2LP 10400683 IC50 = 3.9 nM T99347 D0B4GX 9840951 IC50 > 9100 nM T99347 D0BO6C 4156919 EC50 = 40 nM T99347 D0C0FH 12811063 IC50 = 2.4 nM T99347 D0C2FM 5311462 Ki = 10 nM T99347 D0C6BY 71580330 IC50 = 13 nM T99347 D0C6JG 11333903 IC50 = 589 nM T99347 D0C7TX 16007001 IC50 = 5330 nM T99347 D0C9FH 11615675 IC50 = 1920 nM T99347 D0CQ6I 11608287 Ki = 1.003 nM T99347 D0CT7P 11460152 IC50 = 2300 nM T99347 D0D1GI 10131083 IC50 = 4620 nM T99347 D0D2FB 3361967 Ki = 2100 nM T99347 D0D2GL 3972752 Ki > 1000000 nM T99347 D0D4HG 11245456 EC50 = 10 nM T99347 D0DX6U 23725699 IC50 = 32 nM T99347 D0E3WH 11481793 IC50 = 115 nM T99347 D0E8DM 9881352 IC50 = 140 nM T99347 D0EK6F 16736030 IC50 = 140 nM T99347 D0EK6P 5310984 Ki > 100000 nM T99347 D0F9QY 6604893 EC50 = 2.36 nM T99347 D0G4BW 16659801 IC50 > 1000 nM T99347 D0GA4M 10308060 IC50 = 890 nM T99347 D0GX5C 16725048 IC50 = 10000 nM T99347 D0I6KU 24894087 IC50 = 7.5 nM T99347 D0I9NE 11557579 IC50 = 23 nM T99347 D0IO8J 3025961 IC50 = 2 nM T99347 D0J3NX 44224196 EC50 = 19 nM T99347 D0J4HH 10198811 IC50 = 70 nM T99347 D0JG2W 11381029 IC50 = 320 nM T99347 D0JH2D 11424570 IC50 = 78 nM T99347 D0K0ZK 11383075 EC50 = 157 nM T99347 D0K7KM 44392958 Ki = 10.76 nM T99347 D0L1PQ 10332109 IC50 = 190 nM T99347 D0L2KN 11658509 IC50 = 337 nM T99347 D0L5FW 10910934 IC50 = 1 nM T99347 D0L6PL 16735659 IC50 = 510 nM T99347 D0L9FD 51003564 EC50 = 50.1 nM T99347 D0LP7W 1489963 IC50 = 39.81 nM T99347 D0M2YQ 9967471 IC50 = 6.7 nM T99347 D0N0NJ 15508178 IC50 > 300000 nM T99347 D0N9UZ 9819927 Ki = 8200 nM T99347 D0NB2G 44410045 Ki = 10 nM T99347 D0NS9H 11736483 IC50 = 59 nM T99347 D0OH2P 5311040 Ki = 103000 nM T99347 D0OV2V 6324634 Ki > 300000 nM T99347 D0P0QI 9816778 IC50 = 25 nM T99347 D0P0RY 11535913 Ki = 0.37 nM T99347 D0P2DV 11550292 IC50 = 2966 nM T99347 D0P2IJ 24763119 EC50 = 550 nM T99347 D0P3XO 5311459 IC50 = 155000 nM T99347 D0PN6Z 179394 Ki > 1000000 nM T99347 D0Q6VH 5311432 IC50 = 290 nM T99347 D0QE3C 11379626 EC50 = 14 nM T99347 D0R0IB 56587994 EC50 > 10000 nM T99347 D0R0JE 16735841 IC50 = 6 nM T99347 D0R7VW 11460771 IC50 = 620 nM T99347 D0R8EU 11245287 IC50 = 6200 nM T99347 D0RJ5B 11473392 IC50 = 2860 nM T99347 D0S7SE 10354477 IC50 = 7 nM T99347 D0SB7U 57559562 IC50 = 10000 nM T99347 D0SE2D 23725212 IC50 = 460 nM T99347 D0SF9Z 16118119 IC50 = 4624 nM T99347 D0SG6Q 23634171 IC50 > 3000 nM T99347 D0ST3S 11629906 IC50 = 78.6 nM T99347 D0T4QX 11646823 IC50 = 10 nM T99347 D0T4YQ 16000100 EC50 = 10 nM T99347 D0T7SA 44393041 IC50 = 423 nM T99347 D0TW0I 11715388 IC50 = 3090 nM T99347 D0U0UB 44393020 IC50 = 15 nM T99347 D0U2GG 16736031 IC50 = 4.2 nM T99347 D0V3YX 11537456 IC50 = 147 nM T99347 D0V4RO 10192768 IC50 = 440 nM T99347 D0W0NJ 44442431 IC50 > 100000 nM T99347 D0W1SX 603306 IC50 = 5480 nM T99347 D0W2GG 16659802 IC50 > 1000 nM T99347 D0W5JE 11543200 IC50 = 25.3 nM T99347 D0WJ8I 11708325 IC50 = 654 nM T99347 D0X4UN 966005 IC50 = 5900 nM T99347 D0Y3PV 24777189 EC50 = 1130 nM T99347 D0Z0JU 11321863 IC50 = 138 nM T99347 D0Z0LV 53318624 EC50 = 16 nM T99347 D0Z1PY 11572058 IC50 = 140 nM T99347 D0Z9QZ 44393040 IC50 = 845 nM T16891 D0EV6T 54682461 Ki = 9000 nM T16891 D0CG8S 71305058 IC50 > 200000 nM T16891 D0HM5J 118253852 IC50 > 20000 nM T16891 D04ZIJ 5478883 IC50 = 0.08 nM T16891 D07PSP 5479205 Ki = 142 nM T16891 C7A9BK 65023 IC50 = 2000 nM T16891 CV2P5E 454914 Ki = 90 nM T16891 CX0B5L 9853618 IC50 > 100000 nM T16891 C69KGX 10394329 Ki = 17 nM T16891 C1GYV7 10931081 IC50 = 37.5 nM T16891 CW68BJ 11518143 IC50 > 30000 nM T16891 C5XB3T 11520033 Ki = 2 nM T16891 CE9ZI8 11556254 Ki = 5 nM T16891 C1PSL5 11614083 Ki = 24 nM T16891 C3LW2D 11632240 IC50 = 11000 nM T16891 CLP92O 11963435 IC50 > 30000 nM T16891 CE29TK 14887165 IC50 > 10000 nM T16891 CJO10Z 14887166 IC50 > 10000 nM T16891 C02NGW 14887167 IC50 >> 10000 nM T16891 CJ8R0O 14887174 IC50 = 360 nM T16891 CHIC86 14887175 IC50 = 165 nM T16891 C56EWA 14887177 IC50 ~ 10000 nM T16891 C2LRD8 14887179 IC50 ~ 10000 nM T16891 CT4V6C 14887181 IC50 >> 10000 nM T16891 C4UA0C 14887183 IC50 = 115 nM T16891 C6JF8N 14887185 IC50 = 240 nM T16891 CAKS64 14887194 IC50 ~ 10000 nM T16891 CE12CX 15018069 Ki = 21 nM T16891 CI41XT 15126555 Ki = 0.5 nM T16891 CIV72W 16086657 IC50 = 8100 nM T16891 CMXJ30 23625795 IC50 > 10000 nM T16891 CJUX10 24808497 Ki = 30 nM T16891 CWF5Z3 25143506 IC50 > 30000 nM T16891 C5S6QR 44253975 IC50 = 42.9 nM T16891 CN9BZ7 44253976 IC50 = 0.354 nM T16891 CS7XD5 44321765 Ki = 2 nM T16891 C2OFK8 44321766 Ki = 2.2 nM T16891 CZ45LH 44322035 Ki = 300 nM T16891 CQ09YG 44322074 Ki = 3.3 nM T16891 C3N9LQ 44322075 Ki = 2.9 nM T16891 CK0BQ2 44322083 Ki > 10000 nM T16891 CNT69K 44322084 Ki = 11 nM T16891 CN58AQ 44322086 Ki = 15 nM T16891 C1G0FY 44322087 Ki = 44 nM T16891 CM1HG2 44379569 Ki = 50 nM T16891 C3LA2W 44379720 Ki = 3 nM T16891 CMB9W5 44383534 IC50 = 170 nM T16891 CHL19P 44631842 IC50 = 0.4 nM T16891 C3M7ZG 45105274 Ki = 86 nM T16891 C2YE7A 45254510 IC50 > 1000 nM T16891 C43HDC 45256109 IC50 = 320 nM T16891 CVW76R 46190732 IC50 = 5 nM T16891 CZ0JD1 46191766 IC50 = 4 nM T16891 CM9ON2 46225154 IC50 = 8 nM T16891 C7IJ2F 53232612 IC50 > 10000 nM T16891 C17GML 53465141 IC50 = 75 nM T16891 CAH7Y1 54681312 IC50 > 40000 nM T16891 C3P8YE 54681383 IC50 > 40000 nM T16891 C2TN0J 57379439 IC50 = 0.3 nM T16891 C2PJ4N 59271992 IC50 > 30000 nM T16891 CQW7A8 60149247 Ki = 1100 nM T16891 CUE46I 66575069 IC50 = 36.4 nM T16891 C56CFA 68448803 IC50 > 10000 nM T16891 CTO36I 70680446 IC50 = 9 nM T16891 CDX40V 70680447 IC50 = 210 nM T16891 C9F1QE 70680448 IC50 = 20.8 nM T16891 CDQ09Y 71452058 IC50 = 77.5 nM T16891 CN26XZ 71452059 IC50 = 1710 nM T16891 CA3H9D 71452060 IC50 = 1450 nM T16891 C2UC7A 71452061 IC50 = 30.4 nM T16891 CTV35W 71453879 IC50 = 1520 nM T16891 CLE7P2 71453880 IC50 = 0.724 nM T16891 CO67FA 71453881 IC50 = 1.92 nM T16891 C93BQC 71455611 IC50 = 4.94 nM T16891 CK73LU 71457396 IC50 = 58.2 nM T16891 C1PRD6 71461037 IC50 = 4950 nM T16891 C9L1IU 71461038 IC50 = 51.9 nM T16891 CX34PN 73017594 IC50 = 7050 nM T16891 C72FWD 91929322 Ki = 850 nM T16891 C02GTW 102160610 IC50 = 87000 nM T16891 CELZ36 118866105 IC50 = 1377000 nM T16891 C9M2WU 118866986 IC50 = 453000 nM T16891 CBU0D5 127050883 IC50 = 23 nM T16891 C0JQU4 139589854 IC50 = 100 nM T16891 CF05LW 139589856 IC50 = 0.5 nM T16891 C6HOU5 145950897 IC50 = 5 nM T16891 CU1VE4 145951062 IC50 = 43 nM T16891 C4YMX8 145955472 IC50 = 9 nM T16891 CRA7P1 145958864 IC50 = 23 nM T16891 C2S4ZM 155519404 IC50 = 4000 nM T16891 C7DH9B 155556912 IC50 = 7547 nM T16891 C86SOP 155561681 IC50 = 20000 nM T16891 D0KK6A 15126552 Ki = 0.1 nM T16891 D0P6RT 10078814 Ki = 0.5 nM T16891 D0Y5IQ 44255320 IC50 = 0.8 nM T55916 D0S6QR 214350 EC50 = 2400 nM T55916 D0X7GL 121892 EC50 = 1980 nM T55916 CI1G2C 26873419 IC50 = 200 nM T55916 C7RI0L 66653331 EC50 = 625 nM T55916 C2ORB8 90377311 EC50 = 890 nM T55916 CF0NR7 145981605 EC50 > 10000 nM T55916 CE32VM 145982955 EC50 = 20 nM T55916 CM7TR2 145990268 EC50 = 4000 nM T55916 C94WGB 145990965 EC50 = 160 nM T55916 C52JOD 145993164 EC50 = 100 nM T55916 C30IVC 155491024 EC50 = 100 nM T55916 CTJ34I 155491025 EC50 = 80 nM T55916 C6R4FC 155513238 EC50 = 1420 nM T55916 C12LAI 155521071 EC50 = 2030 nM T55916 C8T4QV 155567226 EC50 = 780 nM T55916 D0N5CH 9903497 EC50 > 10000 nM T55916 D0W2FU 53347902 EC50 > 30000 nM T55916 D0XY2M 3111211 EC50 = 1600 nM T16596 D00IFR 58423153 Ki = 0.23 nM T16596 D07EHV 44814409 Ki = 0.009 nM T16596 D08UUL 46700756 IC50 > 10000 nM T16596 D0E3TC 44259 IC50 = 0.1206 nM T16596 D00OWF 5280953 IC50 = 4300 nM T16596 D04VSB 68356857 IC50 = 4 nM T16596 D06OKX 68356855 IC50 = 2 nM T16596 D06TGF 44479463 IC50 = 440 nM T16596 D08JUU 68327881 IC50 = 5 nM T16596 D0J6HN 46179018 Ki = 0.001 nM T16596 D0M0TH 44480198 IC50 = 200 nM T16596 D0NE0N 44479711 IC50 = 210 nM T16596 D0OS2I 59226518 Ki = 0.003 nM T16596 D0P9UF 51002052 Ki < 3 nM T16596 D09SFV 3973 IC50 = 1400 nM T16596 C5KPL9 977221 IC50 = 4078 nM T16596 C2JSX4 1241442 IC50 = 730 nM T16596 CEW8K1 1379922 IC50 = 390 nM T16596 CWJS81 1539584 IC50 = 280 nM T16596 COPQ34 16043794 Ki = 5.4 nM T16596 C38FDZ 16760660 IC50 = 83 nM T16596 CBG4X2 20784957 Ki = 2900 nM T16596 CP1WR0 24795070 Ki = 24 nM T16596 C4D2QE 24894053 Ki = 0.006 nM T16596 CL85GI 39005031 Ki = 230 nM T16596 CUQE83 44187007 IC50 = 120 nM T16596 C9V3XY 44199470 Ki = 0.02 nM T16596 CU13JS 44217530 Ki < 3 nM T16596 CW96TZ 44217683 Ki = 4 nM T16596 C0LDV8 44222965 IC50 = 57 nM T16596 C3ZJ6S 44222969 IC50 = 35 nM T16596 CPJ3G8 44241505 IC50 = 10 nM T16596 CZ3DI6 44479207 IC50 = 170 nM T16596 CS89EN 44479467 IC50 = 40 nM T16596 CL3M2Q 44545852 IC50 = 16 nM T16596 CEQN62 44609163 IC50 < 3 nM T16596 C7G4FT 44609164 IC50 < 3 nM T16596 CH9FO5 44609165 IC50 < 3 nM T16596 CLPY85 44609168 IC50 < 3 nM T16596 CU0QT2 44609322 IC50 < 3 nM T16596 CQ06VN 44609327 IC50 < 3 nM T16596 CE9GN6 44609485 IC50 = 9 nM T16596 C4QC7B 44609634 IC50 = 42 nM T16596 CDS4J9 46178380 Ki < 3 nM T16596 CP0WY1 46178460 Ki = 14 nM T16596 C4S8MP 46179491 Ki < 3 nM T16596 CLS29B 46872626 IC50 > 10000 nM T16596 C09RXA 46937301 IC50 = 12.4 nM T16596 C04LMP 46937315 IC50 = 90 nM T16596 CPW9Z5 46937316 IC50 = 24 nM T16596 CA18HF 46937317 IC50 = 117 nM T16596 C60WAG 52940742 IC50 = 60 nM T16596 CA3FI5 52943221 IC50 = 6 nM T16596 CR7A0Z 52945651 IC50 = 40 nM T16596 C82IWE 53250611 IC50 = 10600 nM T16596 CNI7P9 53372541 IC50 = 7 nM T16596 C0IYG7 53372543 IC50 = 55 nM T16596 CA6H2P 53372668 IC50 = 16 nM T16596 CY1I9B 53372669 IC50 = 23 nM T16596 COP26H 53372670 IC50 = 40 nM T16596 CFM7W8 53372672 IC50 = 2.5 nM T16596 C9GYZ3 53372790 IC50 = 0.8 nM T16596 C49DRM 53482602 Ki = 0.007 nM T16596 CS4Y9F 53482665 Ki = 0.4 nM T16596 CR9P7C 53482785 Ki = 0.2 nM T16596 C5IWB4 53482960 Ki = 0.2 nM T16596 C2AJ9L 54576042 IC50 = 1.3 nM T16596 CWQ31J 54752779 IC50 = 5 nM T16596 CZ4CR6 54752780 IC50 = 4 nM T16596 C96CIG 54752781 IC50 = 3 nM T16596 C2FK8I 54752782 IC50 < 2 nM T16596 CC7T2A 56674921 IC50 = 100 nM T16596 CFKA67 57390288 IC50 = 490 nM T16596 CYF74P 57390289 IC50 = 14000 nM T16596 C4Y3WA 57390290 IC50 = 5 nM T16596 CU3WM8 57390291 IC50 = 343 nM T16596 CO92HZ 57390346 IC50 = 459 nM T16596 CS0Y1G 57392065 IC50 = 5800 nM T16596 C13ARH 57392066 IC50 = 10000 nM T16596 CG5LM0 57392126 IC50 = 367 nM T16596 C1SGW3 57393817 IC50 = 12000 nM T16596 C34RIH 57393818 IC50 = 310 nM T16596 C29ZPK 57395544 IC50 = 22 nM T16596 CWV27Q 57395545 IC50 = 260 nM T16596 CSZ37K 57396179 IC50 = 3300 nM T16596 C06LDJ 57396331 IC50 = 108 nM T16596 CW4KG3 57396858 IC50 = 28 nM T16596 CIBU80 57397370 IC50 = 12800 nM T16596 CC6Q2N 57397371 IC50 = 5 nM T16596 C1UZP2 57397437 IC50 = 154 nM T16596 C1L4HY 57398127 IC50 = 13 nM T16596 CODG52 57398624 IC50 = 18 nM T16596 C1NLS0 57399688 IC50 = 490 nM T16596 C0YAL9 57399780 IC50 = 235 nM T16596 C4CW2G 57400284 IC50 = 66 nM T16596 CC73VO 57400785 IC50 = 5700 nM T16596 CM7NS6 57400786 IC50 = 6 nM T16596 CX5MH0 57400787 IC50 = 10 nM T16596 CJ4YR1 57400855 IC50 = 235 nM T16596 C36ZSI 57402544 IC50 = 7400 nM T16596 C6F9HJ 57402545 IC50 = 1800 nM T16596 CVBS23 57402546 IC50 = 960 nM T16596 CG35HA 57402547 IC50 < 2 nM T16596 CA71NH 57403845 IC50 = 11 nM T16596 C6JET5 58182164 Ki = 0.19 nM T16596 CXT6Q2 58423155 IC50 = 36 nM T16596 C73BEA 58423187 IC50 = 3200 nM T16596 C3KL4R 58423251 IC50 = 26 nM T16596 CF0L6E 58423275 IC50 < 5 nM T16596 CY2I5D 58423319 IC50 = 5 nM T16596 CBY0I7 58423384 IC50 = 110 nM T16596 CRG4K0 58464982 Ki = 0.009 nM T16596 C6H8IU 59226389 Ki < 3 nM T16596 CCU1I6 59455685 Ki = 4 nM T16596 C9V2EM 60155700 IC50 = 44 nM T16596 C5AQ6G 60155701 IC50 = 130 nM T16596 C1C4BG 60155702 IC50 > 2000 nM T16596 C8SLY4 60168156 IC50 = 41 nM T16596 C57MNF 60168157 IC50 = 200 nM T16596 CFB45M 60168158 IC50 = 80 nM T16596 C4BRH3 62046501 Ki > 12500 nM T16596 CV63UL 67240318 IC50 > 10000 nM T16596 C7FCH0 67959600 IC50 = 5 nM T16596 CB65ES 67959736 IC50 = 1 nM T16596 CE54CI 67960005 IC50 = 142 nM T16596 CY3AZ9 67960061 IC50 = 0.4 nM T16596 CV8O1G 67960139 IC50 = 4 nM T16596 CVFC41 67960161 IC50 = 2 nM T16596 CP2G8D 67960181 IC50 = 0.7 nM T16596 CR7DN8 68032650 IC50 > 1000 nM T16596 CGO14Q 68161034 Ki = 3 nM T16596 C02UIN 68161275 Ki = 20 nM T16596 C4XZ5Q 68161316 Ki = 1000 nM T16596 CA0UR4 68161594 Ki = 5 nM T16596 CY0QN9 68161639 Ki = 490 nM T16596 CD41ZA 68161763 Ki = 50 nM T16596 C0US3B 68161865 Ki = 15 nM T16596 C36FUI 68161871 Ki < 3 nM T16596 CYJQ86 68162030 Ki = 36 nM T16596 C6FEN2 68162062 Ki < 3 nM T16596 CJR94B 68162223 Ki = 21 nM T16596 CAD7C0 68162522 Ki = 5 nM T16596 C9GJN4 68162758 Ki = 180 nM T16596 C09NJI 68162802 Ki < 3 nM T16596 C57KXW 68162851 Ki = 12 nM T16596 C97XLW 68163204 Ki < 3 nM T16596 C1E3XF 68184638 Ki < 3 nM T16596 C3SFB2 68184734 Ki = 3 nM T16596 C9XD8R 68187352 Ki < 3 nM T16596 CH2FV7 68187375 Ki = 0.06 nM T16596 CN6A5W 68187418 Ki < 3 nM T16596 CYM62W 68187421 Ki = 20 nM T16596 CYR6N1 68187478 Ki < 1 nM T16596 C7YX8H 68187480 Ki < 3 nM T16596 CKD38R 68187493 Ki = 3 nM T16596 CU3L1D 68187495 Ki < 1 nM T16596 CY6CG5 68187593 Ki = 5 nM T16596 CUB29K 68187641 Ki = 4 nM T16596 C4VUW2 68328157 IC50 = 18 nM T16596 CA19JZ 68328195 IC50 = 8 nM T16596 CC5F2N 68328262 IC50 = 178 nM T16596 CDP01I 68328283 IC50 = 3 nM T16596 CA1NW4 68328307 IC50 = 1 nM T16596 C2PK9C 68328329 IC50 = 6 nM T16596 CM5NV2 68328390 IC50 = 15 nM T16596 COQ2P8 68328395 IC50 = 11 nM T16596 CRT84L 68328588 IC50 = 5 nM T16596 CGP7B8 68328695 IC50 = 97 nM T16596 C67HDR 68328735 IC50 = 22 nM T16596 C7O9RP 68356711 IC50 = 3 nM T16596 C7GRD4 68356716 IC50 = 2 nM T16596 CYP10F 68356783 IC50 = 186 nM T16596 CQ6VX1 68356838 IC50 = 5 nM T16596 CUKO28 68356850 IC50 = 29 nM T16596 C4JR8X 68356863 IC50 = 181 nM T16596 CT8O2I 69042864 Ki = 0.007 nM T16596 CSD25R 69045198 Ki = 6 nM T16596 C5NL7W 69047229 Ki < 3 nM T16596 CXI31L 69047447 Ki = 90 nM T16596 C6QXP3 69090096 Ki = 3 nM T16596 C7B1IP 69090444 Ki = 3 nM T16596 CRBN93 70687077 IC50 = 500 nM T16596 C5MXU0 70689157 IC50 = 410 nM T16596 C3GDX9 70696694 IC50 = 4 nM T16596 CH7J2X 70982568 IC50 = 0.027 nM T16596 C2WF8G 71202406 IC50 = 257 nM T16596 C4IEN5 71253342 Ki = 0.02 nM T16596 C6VHC3 71253383 Ki = 0.006 nM T16596 C3EF9T 71253391 Ki = 0.016 nM T16596 CQI4F0 71253507 Ki = 1.4 nM T16596 C8NX5J 71253513 Ki = 0.16 nM T16596 C9I2AE 71253517 Ki = 0.68 nM T16596 CTR6B1 71253520 Ki = 6 nM T16596 CP4SE3 71253554 Ki = 0.01 nM T16596 CH9RZ3 71253640 Ki = 0.2 nM T16596 CI4BD1 71253671 Ki = 0.041 nM T16596 CU1QK9 71253681 Ki = 0.07 nM T16596 CZ9DL0 71253684 Ki = 5 nM T16596 CZA1B4 71253727 Ki = 0.12 nM T16596 CDJ29S 71253734 Ki = 0.017 nM T16596 CX7Z3V 71253771 Ki = 0.015 nM T16596 CPLG04 71253796 Ki = 0.037 nM T16596 C8YOC3 71253802 Ki = 4.4 nM T16596 C6QV8R 71253835 Ki = 0.021 nM T16596 CQL89K 71253906 Ki = 0.015 nM T16596 C6YKF5 71253921 Ki = 3.7 nM T16596 CUBE27 71253945 Ki = 9 nM T16596 CP60UQ 71253958 Ki = 0.1 nM T16596 CWRX87 71254005 Ki = 1 nM T16596 CCNF28 71254040 Ki = 5000 nM T16596 CJTH24 71254053 Ki = 115 nM T16596 CW8H0Y 71254055 Ki = 300 nM T16596 C1W5TL 71254066 Ki = 0.29 nM T16596 COM7L3 71254090 Ki = 0.04 nM T16596 CBST91 71254178 Ki = 0.01 nM T16596 C1HB5Q 71254188 Ki = 0.013 nM T16596 C4GTF2 71254199 Ki = 0.2 nM T16596 CB7Z5W 71254288 Ki = 0.1 nM T16596 CA8G2O 71254348 Ki = 0.65 nM T16596 C2CJI8 71254349 Ki = 3.3 nM T16596 C2HKV3 71262574 IC50 = 2 nM T16596 C6RA0F 71262581 IC50 = 7 nM T16596 C9QE2L 71262654 IC50 = 2 nM T16596 C2OA1S 71262676 IC50 = 1 nM T16596 CS3E8P 71262754 IC50 = 1 nM T16596 C90JDF 71262764 IC50 = 1 nM T16596 CP0GU5 71262790 IC50 = 32 nM T16596 CZ89GY 71262793 IC50 = 5 nM T16596 C5DXK1 71307955 Ki = 0.009 nM T16596 C0LI2T 71488479 IC50 = 17 nM T16596 CE41DB 71488550 IC50 = 95 nM T16596 CJR9V5 71488552 IC50 = 80 nM T16596 CT2L4I 71512722 Ki = 400 nM T16596 C1SM3T 71539661 Ki = 0.009 nM T16596 CCN01X 71547862 IC50 = 12 nM T16596 C2P5XS 71580689 IC50 = 470 nM T16596 CZK04P 71580780 IC50 = 119 nM T16596 CR90HX 71580785 IC50 = 546 nM T16596 CW08ZH 71580788 IC50 = 33 nM T16596 C6AN7B 71624486 Ki = 23 nM T16596 CJ4S3H 71624487 Ki = 0.61 nM T16596 CL5SN0 71624488 Ki = 0.053 nM T16596 C06VMT 71624600 Ki = 0.022 nM T16596 CRP0B1 71624601 Ki = 0.14 nM T16596 CEA49N 71624602 Ki = 0.098 nM T16596 CG16LA 71624603 Ki = 0.025 nM T16596 C7AOZ0 71624604 Ki = 0.062 nM T16596 C7L6CY 71624710 Ki = 0.26 nM T16596 CQ8AR2 71624711 Ki = 0.061 nM T16596 CEFO84 71624712 Ki = 0.036 nM T16596 CWK48Z 71624713 Ki = 0.022 nM T16596 CY52PM 71624822 Ki = 0.019 nM T16596 CHW1F2 71723297 IC50 = 210 nM T16596 C4O8YU 71723298 IC50 = 110 nM T16596 CCO28Q 71723299 IC50 = 90 nM T16596 CFS7Y2 71723441 IC50 = 700 nM T16596 COW25I 71723443 IC50 = 100 nM T16596 C97DCN 71723444 IC50 = 110 nM T16596 CCM0S5 71723445 IC50 = 230 nM T16596 C4FU1Q 71723447 IC50 = 600 nM T16596 CPG8H5 71723448 IC50 = 110 nM T16596 C9E4XZ 72546233 IC50 = 1.8 nM T16596 C62JGC 72715291 Ki = 0.02 nM T16596 C6H7QA 72725546 Ki = 140 nM T16596 CJ15KC 72725547 Ki = 220 nM T16596 CQ5K4U 72725607 Ki = 15 nM T16596 CA51GV 73347322 IC50 = 530 nM T16596 C9HTA8 73350405 IC50 = 260 nM T16596 CHZ9U3 73352003 Ki = 0.3 nM T16596 CXZ9J0 73356528 Ki = 0.022 nM T16596 CVF5P0 73603034 Ki = 0.02 nM T16596 CU5K6Q 74983184 Ki = 0.19 nM T16596 CVA40O 74983298 Ki = 0.01 nM T16596 CYRP53 76310130 Ki > 12500 nM T16596 C49LJQ 76317357 Ki > 12500 nM T16596 CXZ30Q 76321071 Ki > 12500 nM T16596 CX4KN2 76331961 Ki = 1500 nM T16596 CXG04C 76331962 Ki = 12000 nM T16596 CJER97 76331963 Ki = 11000 nM T16596 C0AYU9 76335538 Ki = 1700 nM T16596 C28YJW 76335539 Ki > 12500 nM T16596 C24USN 77050662 Ki = 0.008 nM T16596 CROJ27 78103829 Ki = 0.01 nM T16596 CGDC06 86294715 IC50 = 7 nM T16596 C3AF2E 86676680 Ki = 1800 nM T16596 CB7OC1 86681995 IC50 = 0.88 nM T16596 CK8V3O 86725098 IC50 = 267 nM T16596 C5R4CY 87057584 IC50 = 7 nM T16596 C3N2TQ 89914568 Ki = 0.02 nM T16596 CCSB80 90072314 Ki = 0.005 nM T16596 CYW61R 90256619 IC50 = 1 nM T16596 CK79BW 90256983 IC50 = 9 nM T16596 CX8NV6 90257109 IC50 = 185 nM T16596 CX4J8N 90286701 IC50 = 900 nM T16596 C3E6PB 90656756 IC50 = 50.9 nM T16596 C95SGV 90656757 IC50 = 21.7 nM T16596 C0MWE6 90656758 IC50 = 30 nM T16596 CR3J7I 90656759 IC50 = 20.5 nM T16596 CHK6P8 90656760 IC50 = 55.7 nM T16596 CI68DP 90656761 IC50 = 9.9 nM T16596 COC3M0 90656762 IC50 = 31.3 nM T16596 C7JM5Z 90656763 IC50 = 30.2 nM T16596 C3MQ1Z 90656764 IC50 = 7.8 nM T16596 C10XIT 101898720 IC50 = 20 nM T16596 C5N1VZ 102581295 IC50 > 10000 nM T16596 CJ7XB9 118711716 IC50 = 140 nM T16596 CB4GR1 118711717 IC50 = 200 nM T16596 C98LGU 118711718 IC50 = 169 nM T16596 CD18IZ 118711719 IC50 = 400 nM T16596 C0A2RY 118720249 IC50 = 11 nM T16596 C95FJY 118720250 IC50 = 47 nM T16596 C06XZY 118720251 IC50 = 250 nM T16596 CVK71Z 118720252 IC50 = 10 nM T16596 C3CB8J 118720253 IC50 = 5 nM T16596 CV3ZY2 118720254 IC50 = 3400 nM T16596 CNI0U1 118720255 IC50 = 26 nM T16596 CEHY81 118725601 IC50 = 4 nM T16596 C6J7VS 118725602 IC50 = 3 nM T16596 CRY0X4 118725603 IC50 = 14 nM T16596 CTUD48 118725865 IC50 = 4110 nM T16596 C0NE4L 122193063 IC50 = 50 nM T16596 CC7WL9 122193064 IC50 = 26 nM T16596 CZ1NE6 122194258 IC50 = 380 nM T16596 CO3K9M 122194259 IC50 = 600 nM T16596 CI1N4B 122194260 IC50 = 190 nM T16596 CS86FI 122194261 IC50 = 700 nM T16596 C4V5AG 122194268 IC50 = 340 nM T16596 CKR45A 122196350 Ki = 0.013 nM T16596 CIF59P 122196351 Ki = 0.11 nM T16596 C2ES7U 122196352 Ki = 1500 nM T16596 C4I2VM 122196353 Ki = 3100 nM T16596 CZD9W8 123518123 IC50 = 281 nM T16596 C0T6VF 123561371 IC50 = 70 nM T16596 C04QEN 123616291 Ki = 0.01 nM T16596 C7G6IA 123944769 IC50 = 12 nM T16596 CDL2V4 124005596 IC50 = 14 nM T16596 C4ZS6N 127032072 Ki < 3 nM T16596 C1G4ES 127041542 Ki < 3 nM T16596 C8K0WU 127042183 Ki < 3 nM T16596 CU95YJ 127050291 IC50 = 22 nM T16596 CFKY32 129012056 IC50 = 400 nM T16596 C4Q5LF 132471857 IC50 < 3 nM T16596 CGBZ13 134843302 IC50 = 3700 nM T16596 CSNE45 135461314 IC50 = 346 nM T16596 C2UO7P 135566502 Ki = 0.2 nM T16596 CY4D8I 135566504 Ki = 11 nM T16596 C5DOH6 135566645 IC50 = 18 nM T16596 CN6E1U 135566647 IC50 = 11 nM T16596 CH2YR7 135566648 IC50 = 10 nM T16596 CA6EQ3 135856841 Ki < 0.1 nM T16596 CK9M5H 135867902 IC50 = 35 nM T16596 C20HYR 135867903 IC50 = 23 nM T16596 CZ70TA 135867906 IC50 = 13 nM T16596 C0MSR4 135867912 IC50 = 23 nM T16596 CGM17H 135867918 IC50 = 31 nM T16596 CUQ51Z 135867923 IC50 = 30 nM T16596 C0J7RQ 135867925 IC50 = 250 nM T16596 CORN45 135867927 IC50 = 160 nM T16596 CEX54P 135867940 IC50 = 6 nM T16596 C4XA7O 135867941 IC50 = 11 nM T16596 C8MR6U 135867952 IC50 = 1168 nM T16596 C0M9LS 135867953 IC50 = 102 nM T16596 CP1VS6 135867954 IC50 = 810 nM T16596 CIV27R 135867956 IC50 = 166 nM T16596 CN8PW9 135867959 IC50 = 850 nM T16596 CWSI79 135867966 IC50 = 106 nM T16596 CTPK14 135867967 IC50 = 71 nM T16596 CXU39R 135867972 IC50 = 104 nM T16596 C2CZ9L 135867976 IC50 = 21 nM T16596 CDYQ36 135867981 IC50 = 41 nM T16596 CP56XU 135867984 IC50 = 34 nM T16596 C28JUY 135867996 IC50 = 88 nM T16596 C1GBJ8 135867997 IC50 = 8 nM T16596 CC92BK 135867998 IC50 = 17 nM T16596 C6RU2Z 135868002 IC50 = 204 nM T16596 CK2EH9 135921041 Ki = 4 nM T16596 CCV12A 135927921 Ki = 0.7 nM T16596 C1AJ7H 135927923 Ki = 1 nM T16596 CX9SA7 135927946 Ki = 0.3 nM T16596 COM4E6 135927950 Ki = 0.9 nM T16596 CN0J8C 135927973 Ki = 0.3 nM T16596 CG3UZ1 135927974 Ki = 0.4 nM T16596 C1H2EG 135927980 Ki = 43 nM T16596 C14OBQ 135928469 Ki = 0.5 nM T16596 CYTA89 135930672 IC50 = 12 nM T16596 C3YL4I 136042193 IC50 = 875 nM T16596 CS4R2M 136098630 IC50 = 12 nM T16596 CWM2S3 136098631 IC50 = 58 nM T16596 CP3CA4 136189660 IC50 = 5 nM T16596 CC52HL 136189674 IC50 = 4 nM T16596 C4G9BI 136189695 IC50 = 10 nM T16596 CC87DY 136189770 IC50 = 1244 nM T16596 CTL8M5 136189797 IC50 = 8 nM T16596 CX45QN 136189847 IC50 = 11 nM T16596 CTVX09 136189895 IC50 = 20 nM T16596 CFZT23 136189934 IC50 = 8 nM T16596 CV9N1O 136190017 IC50 = 11 nM T16596 CQ85IN 136190059 IC50 = 31 nM T16596 CX8TS5 136190062 IC50 = 9 nM T16596 CLW25G 136190081 IC50 = 286 nM T16596 CAY7U9 136236280 IC50 = 13 nM T16596 C73IGY 136244208 IC50 = 8 nM T16596 CXS5Z6 136254223 IC50 = 5000 nM T16596 C2DNM5 136254224 IC50 > 5000 nM T16596 CQM1U4 136254225 IC50 = 18 nM T16596 COU4C5 136254226 IC50 = 5000 nM T16596 CQU6J7 136254227 IC50 = 4393 nM T16596 CL95WA 136380901 IC50 = 2.5 nM T16596 C4ZEM3 136609604 IC50 = 1.8 nM T16596 C3MK9W 136807986 IC50 > 10000 nM T16596 CVW05E 137175276 IC50 = 18 nM T16596 CXC2B1 137189794 IC50 = 4 nM T16596 CXA14S 137189795 IC50 = 6.4 nM T16596 C3W2XN 137189796 IC50 = 3 nM T16596 CKUP80 137189818 IC50 = 0.8 nM T16596 CJ20SQ 137189865 IC50 = 1.1 nM T16596 CVG90R 137631416 IC50 = 3 nM T16596 CYQJ28 137632388 IC50 = 25 nM T16596 CV1A5N 137633544 IC50 = 492 nM T16596 C6D8IM 137634495 IC50 = 290 nM T16596 CK7QM8 137634713 Ki = 120 nM T16596 CA1D9B 137636162 IC50 = 69 nM T16596 CF65JZ 137636187 IC50 = 0.4 nM T16596 CD5IZ6 137636389 Ki = 0.4 nM T16596 CQ5S9H 137636735 IC50 = 17 nM T16596 C5HD0W 137638179 IC50 = 3 nM T16596 C1MO4H 137638461 IC50 = 6 nM T16596 CUF1D9 137638752 Ki = 0.8 nM T16596 CJ69GR 137638996 IC50 = 12 nM T16596 C30DWC 137642509 Ki = 23 nM T16596 CPO2G4 137642902 IC50 = 28 nM T16596 CHD90A 137643257 Ki = 0.4 nM T16596 C2MO5L 137643556 IC50 = 45 nM T16596 CL6K4E 137643873 IC50 = 1400 nM T16596 C0DAH4 137644542 IC50 = 64 nM T16596 C1H3ZK 137647783 IC50 = 2 nM T16596 C3JDR6 137648580 Ki = 1 nM T16596 CAK39E 137650557 IC50 = 350 nM T16596 CDF3Q7 137650805 IC50 = 400 nM T16596 C8J3RF 137651484 IC50 = 4 nM T16596 CSQG93 137654724 IC50 = 1 nM T16596 CZE82A 137655925 IC50 = 2 nM T16596 CFXC14 137656007 Ki = 0.03 nM T16596 C1BEV7 137656991 IC50 = 27 nM T16596 C72ZDI 137659673 Ki = 0.2 nM T16596 CK03MR 137660117 IC50 = 5620 nM T16596 C4OUD0 137660252 Ki = 270 nM T16596 CW57TM 137661945 IC50 = 480 nM T16596 C07EKN 138454794 IC50 > 10000 nM T16596 CS32YP 145960484 IC50 = 60 nM T16596 CHZ20V 145960670 IC50 = 273 nM T16596 C81DKZ 145960765 IC50 = 11 nM T16596 C8M2RY 145960938 IC50 = 35 nM T16596 CNSO87 145961054 IC50 = 16 nM T16596 CD2O0Q 145961184 IC50 = 29 nM T16596 CY25XU 145961279 IC50 = 26 nM T16596 C8IAB5 145961349 IC50 = 50 nM T16596 CDTI85 145961440 IC50 = 40 nM T16596 CXU40G 145961470 IC50 = 10 nM T16596 CW15YM 145961475 IC50 = 905 nM T16596 CUI86V 145961560 IC50 = 241 nM T16596 CE26LP 145961625 IC50 = 417 nM T16596 CV15YW 145961659 IC50 = 7 nM T16596 C0KY1T 145961724 IC50 = 401 nM T16596 C2YQF0 145961914 IC50 = 69 nM T16596 CH2V4T 145961915 IC50 = 10 nM T16596 CQLA92 145961972 IC50 = 18 nM T16596 COW23H 145962040 IC50 = 30 nM T16596 C7OF6V 145962094 IC50 = 7 nM T16596 CB3O4I 145962109 IC50 = 3050 nM T16596 CP3EH0 145962188 IC50 = 22 nM T16596 C9S8AO 145962192 IC50 = 19 nM T16596 CZIT45 145962335 IC50 = 155 nM T16596 CTN2B1 145962545 IC50 = 183 nM T16596 C5NCH1 145962614 IC50 = 368 nM T16596 C2TRN8 145962743 IC50 = 589 nM T16596 CLS90K 145962852 IC50 = 128 nM T16596 CJD24A 145962897 IC50 = 82 nM T16596 C9C3YP 145962963 IC50 = 247 nM T16596 C69ZIQ 145963064 IC50 > 10000 nM T16596 C01JIP 145963077 IC50 = 877 nM T16596 CJQ78W 145963108 IC50 = 204 nM T16596 CY8RS4 145963277 IC50 = 236 nM T16596 CUI0L7 145963307 IC50 = 137 nM T16596 CO4Y1M 145963467 IC50 = 9 nM T16596 C8QDJ0 145963511 IC50 = 475 nM T16596 C1J5BC 145963517 IC50 = 29 nM T16596 C3TLW0 145963725 IC50 = 33 nM T16596 CYGN68 155510554 IC50 = 82 nM T16596 C2MD1Q 155513187 IC50 > 10000 nM T16596 CDF0I2 155514882 IC50 = 58 nM T16596 C4T6CH 155518837 IC50 = 58 nM T16596 CKD52G 155520766 IC50 = 1550 nM T16596 CJ5L2U 155520986 Ki = 0.02 nM T16596 CM8HF6 155521436 Ki = 0.1 nM T16596 CGQH30 155523583 Ki = 0.01 nM T16596 C3BTZ8 155525211 Ki = 0.005 nM T16596 CE5ZU0 155526194 IC50 = 1 nM T16596 CQ4XA9 155527433 IC50 = 26 nM T16596 C5OBZ9 155527556 Ki = 0.02 nM T16596 C76QNG 155528354 IC50 = 358 nM T16596 C2R8JO 155528784 IC50 > 10000 nM T16596 C2N6XM 155531935 IC50 = 140 nM T16596 C8IP7E 155532982 IC50 = 40 nM T16596 C68GMW 155538446 IC50 > 10000 nM T16596 C9J3IU 155538981 IC50 = 402 nM T16596 CXV14T 155539760 IC50 = 6 nM T16596 C4H0LS 155541271 IC50 = 60 nM T16596 CY8PB1 155542894 IC50 = 238 nM T16596 CE03IU 155543981 IC50 = 4080 nM T16596 CORH39 155553574 IC50 = 300 nM T16596 CH18PL 155553803 IC50 = 55 nM T16596 CZQM57 155554194 IC50 = 735.53 nM T16596 CY6Q8S 155554337 IC50 > 10000 nM T16596 CXO5L1 155556907 IC50 = 6 nM T16596 CU1MA5 155558576 IC50 = 76 nM T16596 CO2I4P 155559898 IC50 = 1800 nM T16596 CG6T9Y 155559978 IC50 = 7 nM T16596 C46LPJ 155563540 IC50 = 131 nM T16596 C13GYL 127031746 IC50 < 5000 nM T16596 D04TPA 72163809 IC50 = 150 nM T16596 D06HVH 54613583 IC50 = 90 nM T16596 D06UKS 44222958 IC50 = 86 nM T16596 D07MQC 9949093 IC50 = 880 nM T82577 D00HDU 91270 IC50 = 2.6 nM T82577 D00SEB 5388962 IC50 = 1.2 nM T82577 D01FJT 656604 IC50 = 7244359.6 nM T82577 D01STB 5362129 IC50 = 4 nM T82577 D03KYG 107807 IC50 = 1.5 nM T82577 D07HGR 5362119 IC50 = 0.1 nM T82577 D0DZ3X 145742 Ki = 86000 nM T82577 D0E6XR 3062316 Ki = 715000 nM T82577 D0I0EG 44093 IC50 = 0.63 nM T82577 D0I7SZ 54892 IC50 = 8.3 nM T82577 D0M5OC 5484727 IC50 = 0.93 nM T82577 D0N5HJ 5462501 IC50 = 1.2 nM T82577 D0N6RF 65999 Ki = 6000 nM T82577 D0Q0PR 54675769 Ki = 167000 nM T82577 D0U2JP 4369359 IC50 = 11000 nM T82577 D0U3EC 5362124 IC50 = 1.7 nM T82577 D09JES 6324648 Ki = 13.8 nM T82577 D0N4IV 10718956 IC50 > 1000 nM T82577 D04MBS 9801007 IC50 = 12 nM T82577 D05NRI 189729 IC50 = 36.31 nM T82577 D05UQD 656629 Ki = 0.015 nM T82577 D06WBA 123742 IC50 = 32000 nM T82577 D0I5QZ 9998020 IC50 = 30 nM T82577 D0K9YR 9810328 IC50 = 2.5 nM T82577 D0T2IQ 443600 IC50 > 100000 nM T82577 CQP46K 3937 IC50 = 3.981 nM T82577 CSH72V 4802 IC50 = 5.012 nM T82577 CXY67D 11163 IC50 = 7244359.6 nM T82577 C43SDH 62956 Ki = 1.5 nM T82577 C7QUA0 71244 IC50 = 3.715 nM T82577 C2N6DR 71320 IC50 = 7 nM T82577 CAM5C0 73086 IC50 = 3801893.96 nM T82577 CZ0M7X 81721 IC50 = 309029.54 nM T82577 C5F9KD 83525 Ki = 50000 nM T82577 C19KSO 85362 IC50 = 10000 nM T82577 C49UDX 88079 IC50 = 1202264.43 nM T82577 C7KR0D 92181 IC50 = 30199.52 nM T82577 CIWS40 92400 IC50 = 0.4 nM T82577 CCOI47 92829 IC50 = 208929.61 nM T82577 CR71YD 92843 IC50 = 2511886.43 nM T82577 C7E9ND 92946 IC50 = 87096.36 nM T82577 C57WLO 92953 IC50 = 602559.59 nM T82577 C2TD8W 96814 IC50 = 190546.07 nM T82577 C3GQ5H 97054 IC50 = 5888436.55 nM T82577 CQL18W 97363 IC50 = 9120108.39 nM T82577 CY23QB 97364 IC50 = 8709635.9 nM T82577 CR01ON 99278 IC50 = 5370317.96 nM T82577 CRE70Y 99978 IC50 = 199.53 nM T82577 C4MKD1 101179 IC50 = 6309573.44 nM T82577 C0WN9F 107994 IC50 = 2.8 nM T82577 CJ1W2Z 108985 IC50 = 229086.77 nM T82577 CP5Q6B 111257 IC50 = 5754399.37 nM T82577 CTM7W0 114973 IC50 = 3.2 nM T82577 CM9S5Q 122113 IC50 = 19.95 nM T82577 CGR1J3 123913 IC50 = 7079457.84 nM T82577 CPIJ02 130842 IC50 = 9400 nM T82577 C0VK5M 133560 IC50 = 1000 nM T82577 CWPS82 133842 IC50 = 1000000000 nM T82577 CRB2Z1 134166 IC50 = 1 nM T82577 C6ZQJ0 137365 IC50 = 31.62 nM T82577 C6XMS5 150903 IC50 = 912010.84 nM T82577 CDCS28 150964 IC50 = 229086.77 nM T82577 C7CN8P 151148 IC50 = 14125375.45 nM T82577 CMY75U 151282 IC50 = 1412537.54 nM T82577 CB3D6T 156271 IC50 = 12 nM T82577 C6TDE7 165505 IC50 = 2818.38 nM T82577 CB9Q1L 168182 IC50 = 1584.89 nM T82577 CLJ9D1 189008 IC50 = 3235936.57 nM T82577 C0R3KO 194156 IC50 = 33113.11 nM T82577 CU0B8E 329113 IC50 = 1096478.2 nM T82577 CJX54Q 335542 IC50 = 10 nM T82577 CP2T7N 443376 IC50 = 220 nM T82577 CO1UK9 444876 IC50 = 128824.96 nM T82577 C9VSE5 446549 IC50 = 10964.78 nM T82577 CZGF79 448982 IC50 = 23 nM T82577 C1BTQ3 494324 IC50 = 12.59 nM T82577 CN67CR 555078 IC50 > 100000 nM T82577 CQ6IO0 1551643 IC50 = 1995262.31 nM T82577 C2AS3C 2724807 IC50 = 4570881.9 nM T82577 CSE85T 2828746 IC50 = 300 nM T82577 C79HSA 2828749 IC50 = 200000 nM T82577 CF47UW 2834684 IC50 = 20 nM T82577 CN52PM 3013625 IC50 = 446683.59 nM T82577 C8SU0O 3033702 IC50 = 0.8 nM T82577 CA6E1H 3080576 IC50 = 5370317.96 nM T82577 C7YDX5 3082827 IC50 = 0.2951 nM T82577 CY36MH 4369380 IC50 = 140 nM T82577 CH01XT 5281656 Ki = 250200 nM T82577 CO58XD 5311161 IC50 > 100000 nM T82577 CF8YR2 5464343 IC50 = 9900 nM T82577 C1YI9C 5464344 IC50 = 1.7 nM T82577 CMAH79 5479774 Ki = 34200 nM T82577 CJHI21 5484352 IC50 = 616595 nM T82577 CF49DL 5490790 Ki = 1.4 nM T82577 CH5U2F 5491963 IC50 = 3801893.96 nM T82577 CF07VG 5496455 IC50 = 457088.19 nM T82577 CTCZ08 5748613 IC50 = 730 nM T82577 C1QBP5 6426706 IC50 = 3235936.57 nM T82577 CV1E8W 6426709 IC50 = 16982436.52 nM T82577 CO03CU 6427013 IC50 = 10000000 nM T82577 C1A6GP 6427052 IC50 = 10000000 nM T82577 C7XIW1 6992396 IC50 = 190546.07 nM T82577 C9W1MN 6992506 IC50 = 10000000 nM T82577 CB5YC3 6992691 IC50 = 7413102.41 nM T82577 CQ5E0R 6992869 IC50 = 1202264.43 nM T82577 CY8UR9 6992873 IC50 = 128824.96 nM T82577 C8Z9OD 6992930 IC50 = 4786300.92 nM T82577 CWC8M3 6993111 IC50 = 1096478.2 nM T82577 CK3Q0Z 6993120 IC50 = 52480.75 nM T82577 C7HIQ9 6998029 IC50 = 2511886.43 nM T82577 CMB48H 7009555 IC50 = 21877.62 nM T82577 C4UO5E 7009596 IC50 = 933254.3 nM T82577 C46LAM 7009644 IC50 = 8511380.38 nM T82577 CH7P4I 7009653 IC50 = 15848.93 nM T82577 C15XOM 7010504 IC50 = 380189.4 nM T82577 C7QV9R 7019085 IC50 = 1995.26 nM T82577 CFW5P0 7020333 IC50 = 457088.19 nM T82577 CP4M1Q 7021854 IC50 = 1995262.31 nM T82577 C36DHQ 7022320 IC50 = 3235936.57 nM T82577 C2PR6I 7023107 IC50 = 3090295.43 nM T82577 CP0BE5 7039484 IC50 = 549540.87 nM T82577 C28NMU 7408195 IC50 = 3715.35 nM T82577 CPU01J 7408255 IC50 = 2300 nM T82577 C5Q9ZO 9601226 IC50 = 1 nM T82577 C02INA 9803222 IC50 = 140 nM T82577 CEX1W2 9822849 IC50 = 87 nM T82577 CDO9J0 9837272 IC50 = 416869.38 nM T82577 CRF51I 9839564 IC50 > 10000 nM T82577 CI7Q0Y 9840601 IC50 = 1400 nM T82577 CZ2HC0 9840687 IC50 = 175 nM T82577 C2MEU1 9844054 IC50 = 52 nM T82577 C38BVX 9870100 IC50 > 1000 nM T82577 C03SVH 9882882 IC50 = 18700 nM T82577 CZ20AN 9905282 IC50 = 12000 nM T82577 C1NDX9 9910508 IC50 = 10000 nM T82577 CVPG59 9932329 IC50 = 35 nM T82577 CVG0O2 9959014 IC50 > 1000 nM T82577 CU61CH 9978465 IC50 = 260 nM T82577 C91HDB 10014925 IC50 = 2300 nM T82577 C8SY5F 10015450 Ki = 126000 nM T82577 C5UH9J 10041763 IC50 = 4 nM T82577 CMD3J1 10047309 IC50 = 4.8 nM T82577 C32OGJ 10071569 IC50 = 25 nM T82577 CH93JG 10093438 IC50 = 460 nM T82577 C63CBL 10107034 IC50 = 11000 nM T82577 CG0DW7 10141595 IC50 > 100000 nM T82577 C05YBI 10336328 IC50 = 10000 nM T82577 CS3ND2 10355231 IC50 = 769000 nM T82577 C5D8ZA 10355232 Ki = 14200 nM T82577 CL73JY 10381547 IC50 = 5000 nM T82577 C4GZ8V 10393285 IC50 = 50 nM T82577 CM0S1U 10426368 IC50 = 16100 nM T82577 CX78MU 10432045 IC50 = 92 nM T82577 CS4G3H 10436816 IC50 > 100000 nM T82577 CU6OH3 10448308 IC50 = 34 nM T82577 CX38EB 10467565 IC50 = 90000 nM T82577 CG6FZ1 10475845 IC50 = 1.698 nM T82577 C9XC8Y 10493383 IC50 = 34000 nM T82577 C4VN0M 10494952 IC50 > 10000 nM T82577 C69RND 10496022 IC50 = 2000 nM T82577 CG32FM 10613145 IC50 > 100000 nM T82577 CQN7S4 10664538 IC50 = 725 nM T82577 C4S3EZ 10710922 IC50 = 1400 nM T82577 CI4SQ2 10732349 IC50 > 100000 nM T82577 CAD84L 10735551 IC50 > 10000 nM T82577 CT78AR 10759255 IC50 = 118 nM T82577 C7O6RU 10759256 IC50 > 10000 nM T82577 CLAP90 10785969 IC50 > 1000 nM T82577 CM74LH 10789594 IC50 > 1000 nM T82577 CFUE14 10829618 IC50 = 8000 nM T82577 C3UCL2 10854279 IC50 = 12400 nM T82577 CKAF49 10900068 IC50 > 1000 nM T82577 CV70TF 10900407 IC50 = 257039.58 nM T82577 CA7B4P 11119038 IC50 = 457.09 nM T82577 C8Q1SZ 11176510 IC50 = 600 nM T82577 CSF91W 11191083 IC50 = 3.8 nM T82577 CC0MU7 11192220 IC50 > 100000 nM T82577 C4ON0L 11442784 IC50 = 72 nM T82577 CE3HA6 11556698 Ki = 0.65 nM T82577 C78VRX 11774785 IC50 = 4000 nM T82577 COT0R7 11792153 IC50 = 22 nM T82577 CJ4VL3 11797382 IC50 > 1000 nM T82577 CSD43L 11989733 IC50 = 20000 nM T82577 C9IG0H 11992410 Ki = 195700 nM T82577 CJK95A 11992491 Ki = 84300 nM T82577 CTL5N6 11992492 Ki = 33600 nM T82577 CSK08P 11992493 Ki = 13300 nM T82577 C6YAP0 11992494 Ki = 43000 nM T82577 CG2ZY3 12190925 IC50 = 1348962.88 nM T82577 C57JAK 12698983 IC50 = 33000 nM T82577 CNU93T 12698984 IC50 = 3700 nM T82577 CRE7O9 12698990 IC50 = 35000 nM T82577 CPE6H9 12698991 IC50 = 30000 nM T82577 CQ6T3P 12698992 IC50 = 19000 nM T82577 C53CVG 12698999 IC50 = 100000 nM T82577 CW3DV9 12785186 IC50 = 67608.3 nM T82577 CC1GB9 12854254 IC50 = 70 nM T82577 CCXB83 12854279 IC50 = 86 nM T82577 C16NQY 12876150 IC50 = 19054.61 nM T82577 C0S2BY 12883918 IC50 = 130 nM T82577 CPV89D 12942866 IC50 = 18 nM T82577 C06PUC 12942868 IC50 = 19.95 nM T82577 CH6GO8 13036940 IC50 = 851.14 nM T82577 CL6T9B 13036944 IC50 = 426.58 nM T82577 C3B6JL 13036947 IC50 = 3019.95 nM T82577 CNU7I4 13044267 IC50 = 300 nM T82577 C58IDW 13044278 IC50 = 3 nM T82577 CGN26M 13069290 IC50 = 100 nM T82577 CDXC29 13104362 IC50 = 72.44 nM T82577 CG4MW9 13105154 IC50 = 1.202 nM T82577 CQT32M 13135337 IC50 = 39.81 nM T82577 CUOP05 13136851 IC50 = 12.59 nM T82577 C2CPA7 13136852 IC50 = 3.981 nM T82577 CCZY61 13144519 IC50 = 2511.89 nM T82577 C83XMT 13144525 IC50 = 1 nM T82577 CQ4DK3 13144530 IC50 = 3162.28 nM T82577 CY05BC 13144539 IC50 = 125.89 nM T82577 C6UFA7 13208321 IC50 = 38904.51 nM T82577 CC9Q7D 13241661 IC50 = 1.995 nM T82577 CD32WB 13335293 IC50 = 39.81 nM T82577 CUOH03 13339952 IC50 = 13 nM T82577 CY6G3M 13375125 IC50 = 3 nM T82577 C1X4KC 13456344 IC50 = 1.7 nM T82577 C3M7TP 13456346 IC50 = 2400 nM T82577 CB2MK0 13456353 IC50 = 5100 nM T82577 CNC8Z9 13456366 IC50 = 1.6 nM T82577 CBA7E6 13456368 IC50 = 2400 nM T82577 CP39OT 13456371 IC50 = 7900 nM T82577 CNW9U6 13456375 IC50 = 1.5 nM T82577 CHE38M 13456380 IC50 = 2.1 nM T82577 C3KAG2 13456384 IC50 = 3.3 nM T82577 CVKP79 13456389 IC50 = 11 nM T82577 CQN8H1 13456394 IC50 = 2.1 nM T82577 CE48FZ 13456399 IC50 = 2.4 nM T82577 CXDK27 13456404 IC50 = 2.3 nM T82577 CK49UY 13456423 IC50 = 6.7 nM T82577 C4TW5G 13477728 IC50 = 2200 nM T82577 C0U9VL 13500748 IC50 = 40 nM T82577 C1WZD8 13500752 IC50 = 15 nM T82577 CF0B3X 13500754 IC50 = 4 nM T82577 C2KD8I 13500765 IC50 = 2.9 nM T82577 C7WFB0 13500770 IC50 = 7 nM T82577 C20UNH 13500773 IC50 = 4 nM T82577 CJUH76 13500778 IC50 = 8.5 nM T82577 CZU08S 13500788 IC50 = 540 nM T82577 C9SL4H 13500790 IC50 = 45 nM T82577 C4VUX3 13500793 IC50 = 1000 nM T82577 CV4DT1 13500795 IC50 = 5 nM T82577 CE04SO 13500798 IC50 = 2600 nM T82577 CX4TI6 13500800 IC50 = 6.5 nM T82577 CGF84D 13500805 IC50 = 6 nM T82577 C4HL9V 13588381 IC50 = 10 nM T82577 C0CY8V 13608313 IC50 = 440000 nM T82577 CW6F9B 13608331 IC50 = 8.1 nM T82577 CY47XT 13652520 IC50 = 10 nM T82577 CW2Y3E 13687301 IC50 = 707.95 nM T82577 CUTA37 13749496 IC50 = 480000 nM T82577 C5WGP2 13749498 IC50 = 19 nM T82577 C69ACG 13749504 IC50 = 10 nM T82577 CUH8T2 14212863 IC50 = 25.12 nM T82577 C81ACD 14212864 Ki = 0.5 nM T82577 CHS29Y 14390729 IC50 = 4 nM T82577 C0N5VL 14540994 IC50 = 200 nM T82577 CZK9D7 14540996 IC50 = 0.5 nM T82577 C8EYH0 14630734 IC50 = 3.236 nM T82577 CO5MX9 14630735 IC50 = 0.4898 nM T82577 CG8S3T 14630739 IC50 = 0.1318 nM T82577 C4IDN0 14630741 IC50 = 338.84 nM T82577 C95DVH 14630745 IC50 = 0.8913 nM T82577 CA59NB 14630749 IC50 = 0.7762 nM T82577 C5GN3K 14630751 IC50 = 0.5248 nM T82577 C3MRF1 14630755 IC50 = 0.5248 nM T82577 C3AV1O 14630757 IC50 = 1.905 nM T82577 C9MA5H 14630761 IC50 = 2.57 nM T82577 CXW6K5 14630765 IC50 = 0.631 nM T82577 CICW62 14630769 IC50 = 0.871 nM T82577 CE1MF9 14630771 IC50 = 15.85 nM T82577 COT04P 14630782 IC50 = 0.2951 nM T82577 CAF28C 14630789 IC50 = 1.072 nM T82577 CYC2U8 14630797 IC50 = 0.2884 nM T82577 CF3TS8 14630801 IC50 = 0.1148 nM T82577 CP73OL 14954082 IC50 = 1995262.31 nM T82577 CLH8D1 15380810 IC50 = 17 nM T82577 CQ20VS 15380813 IC50 = 13 nM T82577 CFX03B 15380816 IC50 = 306 nM T82577 CR40IL 15380817 IC50 = 284 nM T82577 C24BMZ 15380820 IC50 = 4.4 nM T82577 C7R3WN 15380821 IC50 = 28 nM T82577 C93DAN 15615011 IC50 = 2570.4 nM T82577 CQGY31 15838528 IC50 = 33 nM T82577 C9TS8Q 15838530 IC50 = 25 nM T82577 CML3T8 16007169 Ki = 7000 nM T82577 CR0S7G 18542459 IC50 = 1700000 nM T82577 C0SNA2 18601751 IC50 = 10 nM T82577 CSH06N 18608376 IC50 = 7 nM T82577 CFP04Y 18608377 Ki = 11 nM T82577 CGT7B1 20285352 IC50 = 48000 nM T82577 C2YAJ0 20336735 IC50 = 2398.83 nM T82577 C72UNP 20430901 IC50 = 158.49 nM T82577 C1ZUJ8 20430909 IC50 = 63.1 nM T82577 C5YH9C 20430913 IC50 = 125.89 nM T82577 CZ0EC4 20445899 IC50 = 7.943 nM T82577 CZ63YJ 20557515 IC50 = 3.162 nM T82577 CSM6K5 20834249 IC50 = 5.248 nM T82577 CIAR58 21152492 IC50 = 7943.28 nM T82577 C9C3UX 21319418 IC50 = 260000 nM T82577 C7E1XV 21967878 IC50 = 3000 nM T82577 C04LJH 21967881 IC50 = 420 nM T82577 CV8W1T 22799800 IC50 = 64.57 nM T82577 CK6TS0 22805094 IC50 = 229086.77 nM T82577 CSJ07X 22818650 IC50 = 3.7 nM T82577 CF3IS9 22823240 IC50 = 48.98 nM T82577 CU1G0L 22824107 IC50 = 34.67 nM T82577 CFW85M 23322524 IC50 = 4.8 nM T82577 COX68N 23330158 IC50 = 31.62 nM T82577 CBXC05 24424330 IC50 = 0.7 nM T82577 CSWU42 24721360 IC50 = 200 nM T82577 C2MV9X 24882714 IC50 = 1980 nM T82577 CP2LY7 25033280 Ki = 200 nM T82577 C4YKQ1 25033281 Ki = 2700 nM T82577 CR16ZF 25108825 IC50 = 31000 nM T82577 CUC8N5 25141405 IC50 > 100000 nM T82577 CJ0CE4 36688130 IC50 = 6100 nM T82577 C7F3QA 40458146 IC50 = 616595 nM T82577 CT9M6L 40532589 IC50 = 1096478.2 nM T82577 CCH0E2 44266573 IC50 = 3 nM T82577 CXM53J 44266591 IC50 = 7.6 nM T82577 CH7F1P 44266803 IC50 = 1600 nM T82577 CC6SU7 44266804 IC50 = 100000 nM T82577 CY1N3U 44266843 IC50 = 11 nM T82577 CVF0N1 44266856 IC50 = 22000 nM T82577 C6BS5J 44278891 IC50 = 67000 nM T82577 CZ0K4Q 44280449 IC50 = 40.74 nM T82577 CKJ6D4 44288065 IC50 = 13 nM T82577 C1K9TL 44295879 IC50 = 14 nM T82577 C7ZK6W 44295891 IC50 = 36 nM T82577 CSE6U2 44295892 IC50 = 36 nM T82577 CQ07SX 44295893 IC50 = 36 nM T82577 C3G2VM 44295920 IC50 = 183 nM T82577 C6Y1TE 44295939 IC50 = 6.3 nM T82577 C62VIB 44295941 IC50 = 24 nM T82577 CDF39L 44295958 IC50 = 5.4 nM T82577 CFIG72 44295966 IC50 = 14 nM T82577 C6MXZ5 44295979 IC50 = 22 nM T82577 C9F2HK 44296019 IC50 = 18 nM T82577 CD9M3U 44296036 IC50 = 13 nM T82577 C5Z6AR 44296037 IC50 = 31 nM T82577 C0O2CV 44298205 IC50 = 2900 nM T82577 C5D0NQ 44298316 IC50 = 4000 nM T82577 CEU45Z 44298353 IC50 = 4000 nM T82577 CB4PE3 44298355 IC50 = 3600 nM T82577 CJBL20 44298400 IC50 = 4400 nM T82577 CH02UQ 44298401 IC50 = 4000 nM T82577 CL5H7U 44298402 IC50 = 3400 nM T82577 C5G3NH 44298403 IC50 = 800 nM T82577 CUC17Z 44298425 IC50 = 2400 nM T82577 C6WF0X 44298426 IC50 = 3500 nM T82577 CN5A9C 44298428 IC50 = 3500 nM T82577 C14KEU 44298431 IC50 = 2800 nM T82577 CP96RN 44298467 IC50 = 3500 nM T82577 CAQ3R9 44298529 IC50 = 8000 nM T82577 C28WVO 44298544 IC50 = 3800 nM T82577 CB6G8U 44301397 IC50 = 22000 nM T82577 CO53EW 44301408 IC50 = 24000 nM T82577 CGZ1U8 44301409 IC50 > 100000 nM T82577 CC9SL1 44301410 IC50 = 49000 nM T82577 CE9X0Y 44301492 IC50 = 58000 nM T82577 CRB40W 44301493 IC50 = 14000 nM T82577 CJA5G4 44301514 IC50 = 520 nM T82577 CJ75TA 44301544 IC50 = 5.8 nM T82577 C5PY9V 44301552 IC50 = 3.1 nM T82577 CWYK75 44301553 IC50 > 10000 nM T82577 CKX6U5 44301557 IC50 = 58000 nM T82577 C06JQA 44301623 IC50 = 440 nM T82577 CR1M7T 44303110 Ki = 1.3 nM T82577 CW2Y0P 44305060 IC50 = 4900 nM T82577 C73KWG 44305071 IC50 = 50000 nM T82577 CN5YE7 44305121 IC50 = 16 nM T82577 C35AID 44305131 IC50 = 6 nM T82577 CEM4D9 44305132 IC50 = 10 nM T82577 CVS47D 44305140 IC50 = 60 nM T82577 C5D2WT 44305173 IC50 = 20 nM T82577 C45NAZ 44305193 IC50 = 7 nM T82577 CCEN18 44305370 IC50 = 8 nM T82577 C97JBA 44305372 IC50 = 12 nM T82577 CYN2E6 44305391 IC50 = 16 nM T82577 CYU57O 44306009 IC50 = 2398.83 nM T82577 CMC5H9 44314997 Ki = 50000 nM T82577 CNH42V 44316498 IC50 = 30902.95 nM T82577 C31XQM 44316511 IC50 = 645.65 nM T82577 C7BZG0 44316726 IC50 = 1047128.55 nM T82577 CDZ83L 44316727 IC50 = 4570.88 nM T82577 C4R9OS 44316742 IC50 = 389.05 nM T82577 CJC68P 44316752 IC50 = 239883.29 nM T82577 CW7X4R 44316753 IC50 = 3.02 nM T82577 CGS02L 44316769 IC50 = 2.884 nM T82577 CR3U4H 44316777 IC50 = 47863.01 nM T82577 CRS6V0 44316778 IC50 = 8317.64 nM T82577 C0H5KE 44316798 IC50 = 2.884 nM T82577 CO47CU 44316799 IC50 = 100 nM T82577 C9HZU0 44316829 IC50 = 323.59 nM T82577 CD42LH 44316833 IC50 = 77624.71 nM T82577 C5UZ3C 44316834 IC50 = 3467368.5 nM T82577 C90GVY 44316848 IC50 = 2511.89 nM T82577 CF19MI 44316849 IC50 = 12.02 nM T82577 CSJW52 44316850 IC50 = 51.29 nM T82577 CH0R6M 44316851 IC50 = 2.188 nM T82577 C91UJF 44316862 IC50 = 2.188 nM T82577 C9XIC1 44316863 IC50 = 1.096 nM T82577 CSR42L 44316995 IC50 = 218.78 nM T82577 C98RBX 44316996 IC50 = 100 nM T82577 C83GOT 44317006 IC50 = 1819700.86 nM T82577 CET86Y 44317007 IC50 = 758.58 nM T82577 C17PCE 44317014 IC50 = 0.6026 nM T82577 CE0F4B 44317022 IC50 = 15.14 nM T82577 CTPG34 44317023 IC50 = 3.467 nM T82577 CP1ZD0 44317024 IC50 = 0.2512 nM T82577 CREQ84 44317041 IC50 = 38018.94 nM T82577 CP96IH 44317066 IC50 = 2511.89 nM T82577 CLAI57 44317085 IC50 = 25703.96 nM T82577 CFYZ13 44317098 IC50 = 12.02 nM T82577 C97MLC 44317099 IC50 = 2570.4 nM T82577 CV9GO2 44317115 IC50 = 1584.89 nM T82577 CLHB32 44317122 IC50 = 52.48 nM T82577 CP6FN2 44317123 IC50 = 4.786 nM T82577 C90MCR 44317124 IC50 = 0.2291 nM T82577 CM1WH6 44317125 IC50 = 3.02 nM T82577 C63XOZ 44317140 IC50 = 56.23 nM T82577 CUS01W 44317141 IC50 = 436.52 nM T82577 C5Y9TJ 44317145 IC50 = 50.12 nM T82577 C0CQ9A 44317192 IC50 = 4897.79 nM T82577 CQ5F2W 44317193 IC50 = 10232.93 nM T82577 C9LV6D 44317202 IC50 = 64.57 nM T82577 CCK6Q5 44317203 IC50 = 8.913 nM T82577 CE7UV6 44317220 IC50 = 2.57 nM T82577 C05DXW 44317221 IC50 = 63.1 nM T82577 CKDQ56 44317244 IC50 = 2.818 nM T82577 CW5XS4 44317245 IC50 = 645654.23 nM T82577 CL7HU2 44317255 IC50 = 5754.4 nM T82577 CG4MD7 44317265 IC50 = 489778.82 nM T82577 C5VC9Y 44317282 IC50 = 933254.3 nM T82577 CR36KD 44317350 IC50 = 70.79 nM T82577 CYJ4H5 44317359 IC50 = 707.95 nM T82577 CQWT76 44317367 IC50 = 6.457 nM T82577 C43PFU 44321145 IC50 = 12000 nM T82577 COQC17 44321532 IC50 = 1700 nM T82577 C6F5YM 44323100 IC50 = 43 nM T82577 C27WIV 44323101 IC50 = 253 nM T82577 CF2TC5 44323117 IC50 = 42 nM T82577 C2LQX9 44323123 IC50 = 506 nM T82577 CEV4C0 44323191 IC50 = 147 nM T82577 CJW7H8 44323192 IC50 = 18 nM T82577 C6UH2T 44323289 IC50 = 696 nM T82577 CB9PO2 44324428 IC50 > 1000 nM T82577 C3F8DZ 44324530 IC50 = 60 nM T82577 CG6M1Z 44324624 IC50 = 181970.09 nM T82577 CBF46I 44324644 IC50 > 1000 nM T82577 C0Y8EC 44324645 IC50 = 385 nM T82577 CF9M7Y 44324653 IC50 > 1000 nM T82577 CK4R2O 44324830 IC50 = 23 nM T82577 C0O3FJ 44324831 IC50 = 22 nM T82577 C0A8MV 44324877 IC50 = 50 nM T82577 CP6K4X 44325010 IC50 > 1000 nM T82577 C92CXR 44325039 IC50 = 660 nM T82577 CJ6VC5 44325055 IC50 = 100 nM T82577 C9KD1P 44325081 IC50 = 147 nM T82577 C2ZG6V 44325082 IC50 = 414 nM T82577 CE0BW7 44325086 IC50 = 240 nM T82577 C6A1TX 44325087 IC50 = 122 nM T82577 CNHV10 44325092 IC50 = 117 nM T82577 C78HBX 44325093 IC50 = 731 nM T82577 CFNJ58 44325094 IC50 > 1000 nM T82577 CDMZ17 44325095 IC50 = 665 nM T82577 C1V3HD 44325102 IC50 = 65 nM T82577 CNT5D4 44325166 IC50 = 53 nM T82577 C0LH2X 44325169 IC50 = 473 nM T82577 C9ZX5S 44325207 IC50 = 44 nM T82577 CO0S6K 44325221 IC50 > 1000 nM T82577 C24XTA 44325222 IC50 = 138 nM T82577 CX70LB 44325223 IC50 > 1000 nM T82577 CK4XN1 44325232 IC50 = 160 nM T82577 C3J1QZ 44325246 IC50 > 1000 nM T82577 CAI35V 44325247 IC50 = 498 nM T82577 CMZY36 44325303 IC50 > 1000 nM T82577 CSQ37C 44328852 IC50 = 3200 nM T82577 CHA38L 44331702 IC50 = 3.5 nM T82577 CA85MQ 44331737 IC50 = 10000 nM T82577 C0M1RW 44331738 IC50 = 1500 nM T82577 CH8J1T 44336332 Ki = 10 nM T82577 CHD7M2 44337491 IC50 = 5.012 nM T82577 CO6VY1 44337754 IC50 = 3.162 nM T82577 CZ0JK8 44337769 IC50 = 0.7943 nM T82577 C80QCV 44337791 IC50 = 1000000000 nM T82577 CL7K4N 44342229 IC50 > 10000 nM T82577 CC0AG1 44342309 IC50 = 12 nM T82577 CJXP15 44342310 IC50 = 5 nM T82577 C3UHG6 44342481 Ki = 9.8 nM T82577 CEF4J6 44352073 IC50 = 0.6 nM T82577 C6CXD9 44352086 IC50 = 650 nM T82577 C9O7JL 44352389 IC50 = 4200 nM T82577 C4UO8R 44352399 IC50 = 700 nM T82577 C7U0CW 44352420 IC50 = 78000 nM T82577 CXLY79 44352485 IC50 = 16000 nM T82577 C8Q6EW 44358246 IC50 = 2.9 nM T82577 CTE2I6 44358261 IC50 = 8.5 nM T82577 CN0SF8 44358282 IC50 = 5.4 nM T82577 CUY49T 44358403 IC50 = 2600000 nM T82577 CLA34I 44358418 IC50 = 2.9 nM T82577 C2LW8Z 44358438 IC50 = 6 nM T82577 C0KPL6 44358439 IC50 = 9.4 nM T82577 C2EFO5 44364784 IC50 > 10000 nM T82577 CIG7T5 44364906 IC50 = 6000 nM T82577 CF53QE 44364917 IC50 = 470 nM T82577 CM6IJ8 44365196 IC50 = 500 nM T82577 C8D3EI 44365739 Ki = 1.2 nM T82577 C4XOS3 44368279 IC50 = 2400 nM T82577 C89VPA 44368523 IC50 = 90 nM T82577 CA57WU 44368529 IC50 = 260000 nM T82577 CJ4QN7 44368530 Ki = 50000 nM T82577 CBPH20 44368554 IC50 = 0.6 nM T82577 CG75AN 44377126 Ki = 30 nM T82577 CRP20F 44379187 Ki = 1.7 nM T82577 C7EFO1 44383695 IC50 = 6100 nM T82577 C62UTQ 44383743 IC50 = 2800 nM T82577 CTFS09 44384017 IC50 > 10000 nM T82577 CZ9E1G 44384213 IC50 = 4000 nM T82577 CVQ2L3 44384274 IC50 = 4500 nM T82577 CI49UJ 44384300 IC50 = 710 nM T82577 CU87YQ 44384394 IC50 = 300 nM T82577 CRD20Q 44384569 IC50 = 46 nM T82577 C4YK9Q 44384727 IC50 = 10 nM T82577 CVJX47 44384730 IC50 = 15 nM T82577 CJ38IM 44384776 IC50 = 300 nM T82577 C5C9JP 44384800 IC50 = 42 nM T82577 C1GZ3J 44384859 IC50 = 540 nM T82577 CDCY82 44384897 IC50 = 1.4 nM T82577 CQ0CL7 44384992 IC50 = 240 nM T82577 C0W2QL 44384993 IC50 = 5.7 nM T82577 C25WKD 44385190 IC50 = 1300 nM T82577 C2EN3J 44385237 IC50 = 1600 nM T82577 C20YZG 44385438 IC50 = 28 nM T82577 C12UQD 44385469 IC50 = 1.4 nM T82577 CZS79C 44385470 IC50 = 330 nM T82577 CN9YX0 44385527 IC50 = 180 nM T82577 CEI0L8 44385582 IC50 = 1600 nM T82577 C0HDN6 44385628 IC50 = 20 nM T82577 C4YJ6G 44385749 IC50 = 8600 nM T82577 C9XS5C 44385867 IC50 = 25000 nM T82577 C4K1UD 44386281 IC50 = 82 nM T82577 C38FCS 44386286 IC50 = 150 nM T82577 C9XE5J 44386287 IC50 = 4.7 nM T82577 CA3U8H 44386919 IC50 = 656 nM T82577 CF2I3D 44388021 IC50 = 36600 nM T82577 C1FRV0 44400757 IC50 = 14600 nM T82577 CK79BM 44400838 IC50 > 100000 nM T82577 C8J4XB 44401169 IC50 = 31500 nM T82577 CFON28 44404945 IC50 = 0.11 nM T82577 C2PV3I 44404953 IC50 = 5 nM T82577 C6LC0X 44409992 IC50 = 10000 nM T82577 C6T8MR 44415488 Ki = 26300 nM T82577 C06HJB 44446952 Ki = 490 nM T82577 CNK7X5 44446953 Ki = 250 nM T82577 CEB78N 44446954 Ki = 180 nM T82577 CMO78A 44446956 Ki = 570 nM T82577 CV6H2M 44446957 Ki = 410 nM T82577 CF4KE1 44446959 Ki = 1800 nM T82577 CW9C0E 44446960 Ki = 310 nM T82577 CQB5M0 44446963 Ki = 20000 nM T82577 C94POY 44446965 Ki = 1000 nM T82577 CBX2U9 44446967 Ki = 5000 nM T82577 CRZ6B3 44446968 Ki = 1100 nM T82577 CY9O4I 44446969 Ki = 250 nM T82577 C4PQ7D 44446970 Ki = 770 nM T82577 C96KIY 44446972 Ki = 750 nM T82577 CK1EM5 44446974 Ki = 570 nM T82577 C4V6RZ 44446975 Ki = 4000 nM T82577 CBL9E6 44446976 Ki = 950 nM T82577 CVYX54 44446979 Ki = 1800 nM T82577 CAI9Z6 44446980 Ki = 2600 nM T82577 C86KVP 44446984 Ki = 25000 nM T82577 COYX76 44454536 IC50 = 40 nM T82577 CL15BG 44454596 IC50 = 39 nM T82577 CKO40E 44454648 IC50 = 191 nM T82577 C4XKJ6 44454674 IC50 = 23 nM T82577 C9O5YF 44454700 IC50 = 60 nM T82577 C18UOF 44454730 IC50 = 110 nM T82577 CAS59Y 44454780 IC50 = 103 nM T82577 C10OTH 44454833 IC50 = 29 nM T82577 CYK78A 44454905 IC50 = 150 nM T82577 CC2IS3 44454957 Ki = 13000 nM T82577 C1ESI2 44454959 Ki = 620 nM T82577 C8L0MV 44454960 Ki = 700 nM T82577 CBG6T0 44454987 Ki = 200 nM T82577 CN7UW3 44455013 Ki = 9.3 nM T82577 CC5L7S 44455015 Ki = 3400 nM T82577 C6KDT1 44455016 Ki = 8.6 nM T82577 CF4ML7 44455018 Ki = 21 nM T82577 CZI6S1 44455047 Ki = 16 nM T82577 C3UF6E 44455406 Ki = 93 nM T82577 CJG71N 44455407 Ki = 210 nM T82577 C0IR5W 44455428 Ki = 840 nM T82577 C62KSV 44455429 Ki > 10000 nM T82577 CR9WL2 44455430 Ki = 3.2 nM T82577 C6XCJ1 44459080 IC50 = 70000 nM T82577 C31XOD 44459545 IC50 = 110 nM T82577 CR6SJ8 44459614 IC50 = 86 nM T82577 C98LAZ 44459680 IC50 = 14 nM T82577 C1QM5C 44459870 IC50 = 2900 nM T82577 CYTE02 44459897 IC50 = 24 nM T82577 C6XD8J 44459908 IC50 = 220 nM T82577 C15PBV 44461233 IC50 = 290 nM T82577 C25YOU 44461318 IC50 = 3100 nM T82577 CIT5G7 44561891 IC50 > 100000 nM T82577 C90BGR 44561892 IC50 > 100000 nM T82577 C9RGX4 44561893 IC50 > 100000 nM T82577 CU7NP5 44561930 IC50 > 100000 nM T82577 CV21IQ 44561931 IC50 > 100000 nM T82577 CR08WA 44561932 IC50 > 100000 nM T82577 C7H4FK 44581551 IC50 = 100 nM T82577 CM67HS 44581552 IC50 = 250 nM T82577 C2UF1V 44581553 IC50 = 280 nM T82577 CG1VM3 44581554 IC50 = 240 nM T82577 C06ZSJ 44581555 IC50 = 340 nM T82577 C30EFL 44581584 IC50 = 21 nM T82577 CZ4SI2 44581585 IC50 = 210 nM T82577 C4AW6J 44581586 IC50 = 300 nM T82577 CD5EV1 44581587 IC50 = 130 nM T82577 CWI5O1 44581588 IC50 = 280 nM T82577 CL98VN 44581589 IC50 = 4000 nM T82577 CV8CA3 44581623 IC50 = 100 nM T82577 CGOQ13 44581624 IC50 = 260 nM T82577 CH3J8K 44581625 IC50 = 340 nM T82577 C87OUW 44581626 IC50 = 370 nM T82577 CA1TE8 44581627 IC50 = 4600 nM T82577 C9LHM3 44581628 IC50 = 300 nM T82577 CXK2B6 44581658 IC50 = 320 nM T82577 CBZ2Y9 44581659 IC50 = 300 nM T82577 C9DEN6 44581660 IC50 = 300 nM T82577 C8FSX4 44581661 IC50 > 10000 nM T82577 C75IKN 44581662 IC50 = 200 nM T82577 CEF4P5 44581663 IC50 = 340 nM T82577 CV6U4W 44581700 IC50 = 430 nM T82577 CF2YX7 44581701 IC50 = 3600 nM T82577 CFR07N 44581702 IC50 = 1700 nM T82577 CBZ8Q9 44581703 IC50 = 260 nM T82577 C7EK0V 44581746 IC50 > 10000 nM T82577 CL1X5R 44586759 IC50 = 2.4 nM T82577 CEB7D9 44586760 IC50 = 0.18 nM T82577 CMZ46U 44586761 IC50 = 0.029 nM T82577 CXL2R9 44586792 IC50 = 3.2 nM T82577 C9ZCP2 44586816 IC50 = 4.2 nM T82577 C3TN5U 44586817 IC50 = 8.4 nM T82577 CY3OW4 44586818 IC50 = 19 nM T82577 CY4A5N 44586819 IC50 = 15 nM T82577 CH5I4V 44586820 IC50 = 0.9 nM T82577 CMN6G9 44586856 IC50 = 2.3 nM T82577 CRE49N 44586857 IC50 = 4.1 nM T82577 CQAG69 44586858 IC50 = 410 nM T82577 CJA8U3 44586859 IC50 = 280 nM T82577 CQ8T1C 44586860 IC50 = 3.3 nM T82577 CA1YC9 44626604 Ki = 1.4 nM T82577 CK6S5H 44626708 Ki = 3.6 nM T82577 C0EJ1F 44626709 Ki = 0.4 nM T82577 CZR23J 44626710 Ki = 3.8 nM T82577 CQB06H 44626711 Ki = 0.41 nM T82577 C17IGS 44627959 Ki = 13 nM T82577 CM1DL3 44627960 Ki = 5 nM T82577 CNZ8L0 44628063 Ki = 20 nM T82577 CRU86P 44628064 Ki = 25 nM T82577 CS5BG9 44628065 Ki = 12 nM T82577 C65RAJ 45102601 IC50 > 10000 nM T82577 C03HVM 45267758 IC50 = 830 nM T82577 CJ73YP 45267767 IC50 = 160 nM T82577 CG80EY 45269496 IC50 = 280 nM T82577 CT15VE 45270333 IC50 = 400 nM T82577 C48XKY 45272068 IC50 = 300 nM T82577 CX4DS1 45273826 IC50 = 1010 nM T82577 CTOA14 45485236 Ki = 16 nM T82577 CJH50R 49797481 IC50 > 100000 nM T82577 CN12AO 53353383 IC50 = 158 nM T82577 C51GUC 53354365 IC50 = 51 nM T82577 CRJ5P9 53354369 IC50 = 279 nM T82577 C4G2HT 53354470 IC50 = 8.6 nM T82577 C9NE6D 54039314 IC50 = 7.7 nM T82577 CR8M4Y 54082602 IC50 = 17 nM T82577 CCRF59 54268836 IC50 = 330000 nM T82577 CU92WO 54311655 IC50 = 2 nM T82577 C6KH4Z 54395218 IC50 = 700 nM T82577 CBGY97 54468999 IC50 = 44 nM T82577 CO8BM6 54560245 IC50 = 3 nM T82577 C2L5QR 54587395 Ki = 0.16 nM T82577 CGH0S7 54589400 IC50 > 100000 nM T82577 C3S0IT 57393223 IC50 = 580 nM T82577 CC2P9X 57394944 IC50 = 140 nM T82577 CF54YD 57396692 IC50 = 220 nM T82577 CDFA84 57396694 IC50 = 460 nM T82577 C2QE1B 57396695 IC50 = 4800 nM T82577 CA2D6Y 57398463 IC50 = 2000 nM T82577 C3OR9M 71449055 IC50 = 40 nM T82577 C2JE4T 71449056 IC50 = 1400 nM T82577 CUG54A 71454428 IC50 = 4.8 nM T82577 CF6S3Y 71456660 Ki = 3 nM T82577 CY6L9B 71459996 IC50 > 1000 nM T82577 CMF80T 71461712 IC50 = 1100 nM T82577 C4FWY1 71462052 IC50 = 12 nM T82577 C3PU7K 71718514 IC50 = 1.2 nM T82577 C1CKV6 71750764 IC50 = 90000 nM T82577 CA29QZ 72697595 IC50 = 40 nM T82577 CT2MS6 72697596 IC50 = 30 nM T82577 CJXR64 90655798 Ki = 21 nM T82577 CXP0U7 90655799 IC50 = 52 nM T82577 C0XQW8 90655800 IC50 = 220 nM T82577 C54ESG 90668209 IC50 > 31622.78 nM T82577 CX4MK8 90668210 IC50 > 31622.78 nM T82577 CX5MA6 90668211 IC50 > 31622.78 nM T82577 C3YZO5 90668278 IC50 > 31622.78 nM T82577 C8LC4Z 118718824 IC50 = 92 nM T82577 CC80MR 122179189 IC50 = 113000 nM T82577 C2A7DH 122179190 IC50 = 347000 nM T82577 C9QKI3 127020966 IC50 > 100000 nM T82577 CJ98CG 132451821 Ki = 7400 nM T82577 CJZ9I0 145949262 IC50 = 460000 nM T82577 CXE5B0 145949765 IC50 = 2.846 nM T82577 C3P4CF 145951239 IC50 = 7.64 nM T82577 CG1W2X 145951970 IC50 = 9.82 nM T82577 C8WMN6 145952431 IC50 = 11.8 nM T82577 CQ35SP 145953190 IC50 = 10.67 nM T82577 CVUC48 145953329 IC50 = 24.22 nM T82577 CXY8W2 145953611 IC50 = 18.97 nM T82577 C6MTC3 145957046 IC50 = 22.3 nM T82577 C5D9GN 145958042 IC50 = 15.11 nM T82577 CE41NM 145958358 IC50 = 112 nM T82577 CA7YZ0 145959902 IC50 = 4.11 nM T82577 CE72UY 145963315 IC50 = 8.841 nM T82577 C7JFL1 145984090 IC50 = 43 nM T82577 CFXM92 145994098 IC50 = 2100 nM T82577 CU42CE 155567829 IC50 > 100000 nM T82577 D00KEP 6049 IC50 = 14000 nM T82577 D02BTV 9816867 IC50 > 100000 nM T82577 D02FMN 9827219 Ki = 7 nM T82577 D02NQB 10430040 IC50 > 100000 nM T82577 D03QJA 11718722 IC50 = 193 nM T82577 D03SPJ 73568 IC50 = 3700000 nM T82577 D03UIF 9906720 IC50 = 520 nM T82577 D07APP 131255 IC50 = 13400 nM T82577 D08ELY 9838786 IC50 = 81000 nM T82577 D0A1CM 5281855 IC50 = 5000000 nM T82577 D0B3UN 44580458 Ki > 100000 nM T82577 D0C6QS 3001497 IC50 = 400000 nM T82577 D0G3YZ 11391583 IC50 > 250000 nM T82577 D0K0OY 44346192 Ki = 100 nM T82577 D0N4RO 44377139 Ki = 520 nM T82577 D0N6CD 10565532 IC50 > 100000 nM T82577 D0N8YA 159596 IC50 > 100000 nM T82577 D0PB5Q 3132 IC50 = 316.23 nM T82577 D0Y3TZ 370 IC50 = 7700000 nM T82577 D0Y5IQ 44255320 IC50 = 10000 nM T98798 CW07XZ 9935056 IC50 > 3300 nM T98798 C3KRX9 23107452 IC50 = 150 nM T98798 C6YH4P 134159047 IC50 > 25000 nM T98798 C0W5RC 145951177 IC50 > 19000 nM T98798 C7TK8Y 145952237 IC50 > 25000 nM T98798 C20JWU 145955054 IC50 > 60000 nM T98798 CVN27T 145955276 IC50 > 25000 nM T98798 CG5D9F 145957954 IC50 > 25000 nM T98798 C5ID6C 145959335 IC50 > 24000 nM T98798 C3LO4I 145959572 IC50 > 25000 nM T98798 CG1O5P 145959656 IC50 > 25000 nM T98798 CJ08IV 145973619 IC50 > 25000 nM T92072 D05DVP 5717 IC50 > 10000 nM T92072 D06ACW 6083 EC50 = 500 nM T92072 D06IAR 60961 IC50 = 2.344 nM T92072 D09AMZ 1676 Ki = 42000 nM T92072 D0B3HD 2519 Ki > 10000 nM T92072 D0F8RA 2153 Ki = 0.6 nM T92072 D0H3WI 37542 Ki = 7410 nM T92072 D0R4UW 449193 IC50 > 1000 nM T92072 D0X3FX 5284596 Ki > 50000 nM T92072 D0XE1C 219024 Ki = 3770 nM T92072 D00OAU 9869857 Ki = 369 nM T92072 D00SUK 216466 Ki = 7 nM T92072 D02OZK 11404337 Ki = 5000 nM T92072 D02YQO 10668061 Ki = 1.111 nM T92072 D03OQI 11618368 Ki = 1350 nM T92072 D05KBP 11610599 Ki = 0.97 nM T92072 D06MIQ 9910098 Ki = 10000 nM T92072 D07TEP 10117987 Ki = 295 nM T92072 D09TFB 9896267 IC50 = 5200 nM T92072 D0F4ZY 5311037 Ki = 841 nM T92072 D0F5UN 9953065 Ki = 1 nM T92072 D0G4CF 11270783 Ki = 1940 nM T92072 D0I3YX 9936489 EC50 = 0.1 nM T92072 D0L5VS 6448585 Ki > 10000 nM T92072 D0QG9A 9805430 Ki = 77 nM T92072 D0U0KR 3035850 Ki = 5.26 nM T92072 D0X0IY 64627 Ki = 0.295 nM T92072 D0Y6ZK 123683 Ki = 3.73 nM T92072 D0Z3PO 21874557 Ki = 68 nM T92072 D0Z9RJ 11561692 Ki = 12 nM T92072 D08ECB 11716665 Ki > 1000 nM T92072 D0I5VA 11248240 Ki = 260 nM T92072 D00YSJ 158795 Ki = 2.05 nM T92072 D01VPK 6439091 Ki = 0.4898 nM T92072 D07ESH 176408 Ki = 287 nM T92072 D0EK6D 3035594 Ki = 12 nM T92072 D0J2UW 3086599 Ki = 289 nM T92072 D0NQ5I 65710 Ki = 39 nM T92072 D0V5DX 9884817 Ki = 3.89 nM T92072 D0Y6GJ 176407 Ki = 178 nM T92072 C7B8VJ 44405080 Ki = 18.3 nM T92072 CF92BM 45482610 EC50 = 8.2 nM T92072 CR04HC 5480 EC50 = 10300 nM T92072 C6GN7M 40692 Ki = 14044 nM T92072 C6MK3J 41211 EC50 = 440 nM T92072 CKF52M 71593 Ki > 100000 nM T92072 CA9Z0E 78268 Ki = 270 nM T92072 C4DG1O 94136 EC50 = 490 nM T92072 C3SPQ5 95121 Ki > 100000 nM T92072 C2CG8M 98567 Ki = 36.7 nM T92072 CGB03T 102175 Ki = 6000 nM T92072 CC90DA 102213 EC50 > 3000 nM T92072 CMT4D5 104924 Ki > 10000 nM T92072 C57IVM 126054 Ki = 10.4 nM T92072 CGA17S 127779 IC50 > 100000 nM T92072 C6OGM1 131432 Ki = 221 nM T92072 CV57OH 131584 Ki = 10.5 nM T92072 C6X3WZ 133012 IC50 = 10 nM T92072 CU7A5O 149362 IC50 = 112 nM T92072 CB6K2R 184691 Ki = 2.5 nM T92072 CL08HI 185566 Ki > 100000 nM T92072 CLQ01J 207319 EC50 > 20000 nM T92072 CQGD08 212359 EC50 = 11700 nM T92072 CA6E5H 215492 Ki = 12.8 nM T92072 CD0MT5 215610 Ki = 27 nM T92072 CA8H6D 264296 EC50 > 20000 nM T92072 CMH1F9 308531 Ki = 23 nM T92072 C5BK1O 314836 Ki > 10000 nM T92072 CVD90Q 377427 Ki = 15.85 nM T92072 C5X4WC 386673 Ki = 10000 nM T92072 CLZE79 386674 Ki = 299 nM T92072 C7SG9U 386679 Ki = 1995.26 nM T92072 CW4FT7 395949 Ki = 398.11 nM T92072 C58QWF 456309 Ki = 244 nM T92072 C9GZ0J 541903 Ki = 1660 nM T92072 C4Y0MB 562794 EC50 = 15200 nM T92072 CI0CW2 570244 Ki = 1900 nM T92072 CE9CN4 571407 Ki = 23 nM T92072 C07HST 608239 Ki = 3981.07 nM T92072 CI1S8O 611038 EC50 > 20000 nM T92072 CX31PR 621302 Ki = 2200 nM T92072 CSV78R 626711 Ki > 100000 nM T92072 CXI3Y4 645569 Ki = 75857.76 nM T92072 CWT5D4 647821 EC50 = 13600 nM T92072 C7HKX6 658709 Ki = 86 nM T92072 C03TBX 679358 Ki = 74.13 nM T92072 C91KES 682802 EC50 = 2800 nM T92072 C2HTM9 686655 Ki = 865 nM T92072 C5FEO8 700373 Ki = 510 nM T92072 C6HF1U 700447 EC50 = 11200 nM T92072 C5X7WA 711464 Ki = 192 nM T92072 C3FHO2 719449 EC50 = 4300 nM T92072 CLT4W1 723688 Ki = 900 nM T92072 C43MFG 737136 EC50 = 3950 nM T92072 CZ6R2E 747391 Ki = 95 nM T92072 C3VO0F 791098 Ki = 7 nM T92072 CJW1K9 828537 Ki = 36 nM T92072 C8Y4NV 851050 Ki > 10000 nM T92072 CC94MT 851051 Ki > 10000 nM T92072 CCM2J1 851052 Ki > 10000 nM T92072 C0VHM4 852929 Ki < 100000 nM T92072 CEQ6K1 852941 Ki = 22908.68 nM T92072 CNJC61 853426 Ki = 7.2 nM T92072 CC1M8O 856282 Ki = 66 nM T92072 CE16YW 856297 Ki = 94 nM T92072 C50HPR 856323 Ki = 42 nM T92072 C9ZKY0 861990 Ki = 2060 nM T92072 CHJV30 906099 Ki > 1000 nM T92072 C1WHL8 916396 Ki = 239 nM T92072 C7YQ1A 917384 Ki = 59 nM T92072 C5QFM2 933735 Ki = 5000 nM T92072 CBS70C 1069525 Ki = 6918.31 nM T92072 CV79ER 1350383 Ki = 208.93 nM T92072 C5P2TF 1487654 Ki > 10000 nM T92072 CI5J9A 1487656 Ki > 10000 nM T92072 CM80QJ 1509337 Ki = 220 nM T92072 CO7S1B 1532293 Ki = 400 nM T92072 C1TV4B 1618253 Ki = 25703.96 nM T92072 CVY75G 1897979 EC50 = 11600 nM T92072 CW2H9O 1898787 Ki = 108 nM T92072 CLU5E8 1899510 Ki = 175 nM T92072 CEJX51 2147018 Ki = 19952.62 nM T92072 C1G8JF 2288678 EC50 = 2700 nM T92072 CD5A1B 2727500 EC50 = 9750 nM T92072 CK8T0W 2748282 Ki > 10000 nM T92072 CRB27T 2763861 EC50 > 20000 nM T92072 C4P8VN 2794740 EC50 = 13200 nM T92072 C4Q5ZI 2814020 EC50 > 20000 nM T92072 CD84EF 2817023 Ki = 29 nM T92072 C51GNW 2874872 Ki > 10000 nM T92072 CHWU72 2910343 Ki > 100000 nM T92072 CS6Q9H 2989397 Ki > 100000 nM T92072 CRO73B 2989630 Ki = 16700 nM T92072 C9UYC2 3000506 Ki = 1221 nM T92072 C80EBV 3000516 Ki = 8607 nM T92072 C5TCF2 3044933 Ki = 12 nM T92072 CC48UQ 3162481 Ki = 10000 nM T92072 CPNR09 3162488 Ki > 10000 nM T92072 C4ZI9K 3162667 Ki > 1000 nM T92072 CSVD14 3349998 Ki = 15 nM T92072 C9Y3AH 3663377 Ki = 18620.87 nM T92072 CSR1K4 3751417 Ki = 1744 nM T92072 CUE3C9 4382765 Ki > 10000 nM T92072 CWP4O1 4412077 Ki > 10000 nM T92072 C7WLX1 4440797 EC50 > 20000 nM T92072 CKH03U 4480217 Ki > 10000 nM T92072 CQGM94 4897338 Ki = 3235.94 nM T92072 C1H4NC 5014044 Ki = 1122.02 nM T92072 C70ILQ 5033052 Ki = 54.3 nM T92072 CZB37F 5311431 Ki = 0.38 nM T92072 C25LIE 5373676 Ki = 7943.28 nM T92072 C80UKF 5467768 Ki = 5.012 nM T92072 CX43YD 5468910 Ki = 5.012 nM T92072 CL9PK8 5516328 Ki = 13489.63 nM T92072 CC0P2D 6032251 Ki = 2511.89 nM T92072 CTK1P2 6439089 Ki = 140 nM T92072 CU6KF1 7162129 Ki = 1258.93 nM T92072 CKP71E 8379104 Ki = 6165.95 nM T92072 C3O8GK 9247074 Ki = 6500 nM T92072 C32LEZ 9497523 Ki = 28 nM T92072 C3M2KJ 9795907 EC50 = 9800 nM T92072 CSN3H2 9798222 Ki = 0.45 nM T92072 C7BR3G 9799990 EC50 = 31.2 nM T92072 CKNT38 9801343 Ki = 1097 nM T92072 CRHL94 9803956 Ki > 4000 nM T92072 C2EJD7 9803992 Ki > 10000 nM T92072 C92LUT 9805713 Ki = 35 nM T92072 C98ERU 9814428 Ki = 26.2 nM T92072 CM96GZ 9814538 Ki = 254 nM T92072 CF8V3M 9818556 Ki = 284 nM T92072 C0JI5S 9819926 Ki = 25.12 nM T92072 CVLM89 9821879 Ki = 76 nM T92072 C1MN3A 9821924 Ki = 2300 nM T92072 C0TS3U 9822488 Ki = 990 nM T92072 C2O9IQ 9822747 Ki = 350 nM T92072 CAQS87 9824812 Ki = 796 nM T92072 CK0FX6 9825550 Ki = 40.1 nM T92072 CG0J6I 9825790 Ki = 137 nM T92072 CUG62V 9827467 Ki = 161 nM T92072 CNM9W5 9828356 Ki = 7300 nM T92072 CFLM79 9834242 Ki = 3624 nM T92072 CLMN73 9834888 Ki = 1273 nM T92072 CTGU01 9835359 Ki = 57 nM T92072 C9BZC8 9836304 Ki = 1665 nM T92072 CS6IN9 9839378 Ki = 20 nM T92072 CFXZ58 9839545 Ki = 94.6 nM T92072 CVG2K1 9839953 EC50 = 2600 nM T92072 C4TOH3 9841364 Ki = 20 nM T92072 C25KVI 9842054 Ki = 14 nM T92072 C12UDF 9843101 Ki > 10000 nM T92072 CKZ07C 9843424 Ki = 251.19 nM T92072 CU6Q8E 9844060 Ki = 9 nM T92072 CUYI26 9844693 Ki = 9.6 nM T92072 CJ8LT7 9848518 IC50 > 10000 nM T92072 CRLO45 9850648 Ki = 136 nM T92072 C2F8KA 9850900 Ki = 690 nM T92072 C3MDK9 9856035 Ki = 10.4 nM T92072 CKEA76 9856296 Ki = 17 nM T92072 CUB8T7 9857266 Ki = 1117 nM T92072 CUZL86 9857422 Ki = 78 nM T92072 CP50JH 9857698 Ki = 45 nM T92072 CUO04X 9857735 Ki = 63 nM T92072 CVR73U 9857814 Ki = 1444 nM T92072 C52DIU 9858247 Ki = 519 nM T92072 CYXI30 9858577 Ki = 894 nM T92072 C6IK1X 9858578 Ki = 553 nM T92072 CUGV50 9860013 Ki = 207 nM T92072 CZRS26 9863617 Ki = 1330 nM T92072 CTK0Z8 9865923 Ki > 6000 nM T92072 CZN45Y 9865975 Ki = 467 nM T92072 CV19SJ 9868763 Ki = 300 nM T92072 CRJ04W 9868991 Ki = 352 nM T92072 C7ARK4 9870396 Ki = 1200 nM T92072 CT2C6K 9870702 IC50 > 10000 nM T92072 CQR53Y 9870718 Ki = 335 nM T92072 CG47TN 9870719 Ki = 234 nM T92072 C36IFS 9879687 Ki = 264 nM T92072 C1ZH7A 9880379 Ki = 984 nM T92072 CQ0T4V 9880392 Ki = 154 nM T92072 CYPJ74 9880921 Ki = 400 nM T92072 C5URA3 9881967 Ki > 10000 nM T92072 CB26YS 9883190 Ki = 2640 nM T92072 CL6AW0 9886589 Ki = 33 nM T92072 CZN50C 9887859 Ki = 250 nM T92072 CLIE16 9890003 Ki = 1015 nM T92072 C7C5VN 9890439 Ki = 160 nM T92072 C8LSD7 9893136 Ki = 65 nM T92072 CE5G7X 9900111 Ki = 1260 nM T92072 CF6M1U 9900245 Ki = 908 nM T92072 C7AE0U 9901099 Ki = 252 nM T92072 CCI2A0 9901100 Ki = 1083 nM T92072 C0RCP7 9901171 Ki = 131 nM T92072 CDPV97 9901196 Ki = 314 nM T92072 CW8PY4 9901260 Ki = 105 nM T92072 CJKD76 9901497 Ki = 132 nM T92072 CW8Z9K 9901700 Ki = 77 nM T92072 CMKV90 9901760 Ki = 12 nM T92072 CCJ95I 9902054 Ki = 1.7 nM T92072 CTU57Q 9902350 IC50 > 10000 nM T92072 CA52RY 9902562 Ki = 86 nM T92072 CJ3OC1 9902563 Ki = 203 nM T92072 CE4G3C 9903342 Ki = 181 nM T92072 C7YM0O 9904456 Ki = 8.4 nM T92072 CF54HI 9904688 Ki = 709 nM T92072 CUG70S 9906178 EC50 = 21.5 nM T92072 CR4SN0 9910158 Ki = 249 nM T92072 CDN1R5 9910926 Ki = 30 nM T92072 C37VQP 9911385 Ki = 49 nM T92072 CC9FE0 9912816 Ki = 54.7 nM T92072 CUM73L 9921668 Ki = 240 nM T92072 CO9WC2 9922606 Ki = 23000 nM T92072 CMGL57 9923269 Ki = 170 nM T92072 CO7FP5 9924271 Ki = 3780 nM T92072 C8CU7X 9924272 Ki = 1760 nM T92072 CO52VW 9924325 Ki = 2090 nM T92072 CLK76N 9924994 Ki > 10000 nM T92072 CA4OK7 9925574 Ki = 303 nM T92072 CXWU86 9929340 Ki = 12.9 nM T92072 CDQN01 9929405 Ki = 15 nM T92072 C7X1TD 9929470 Ki = 594 nM T92072 C1R8JD 9930130 Ki = 66 nM T92072 C8TMY5 9932840 Ki = 2.7 nM T92072 CJ5YV8 9935943 Ki = 161 nM T92072 CO3MX7 9935978 Ki = 30.1 nM T92072 CY82JD 9936058 Ki = 3030 nM T92072 CR05XW 9936467 Ki = 225 nM T92072 CJCR41 9944894 Ki = 17 nM T92072 CW4NR7 9945226 Ki = 76 nM T92072 CD4SZ1 9945283 Ki = 1630 nM T92072 CL3MY6 9946338 Ki = 4.52 nM T92072 CBZG96 9949541 Ki = 17 nM T92072 C1VU2P 9949650 Ki = 25 nM T92072 C4MSO1 9950776 Ki = 2 nM T92072 C9F7BL 9953799 Ki = 1026 nM T92072 CS23VQ 9954406 Ki = 29 nM T92072 C2KD6M 9954747 Ki = 141 nM T92072 C8WR2V 9955052 Ki = 392 nM T92072 C7GH6I 9957239 Ki = 4890 nM T92072 CE0N2P 9965093 Ki = 413 nM T92072 CE3O1U 9966890 Ki = 1680 nM T92072 CND8Q6 9967146 Ki = 130 nM T92072 CO1NR5 9967147 Ki = 612 nM T92072 CPGT28 9967620 Ki = 231 nM T92072 C2UF7H 9968253 Ki = 105 nM T92072 CDM42Y 9970296 Ki = 45 nM T92072 CMZ6X7 9970667 Ki = 62 nM T92072 CNE43U 9970832 Ki = 3.2 nM T92072 CH5XN6 9972895 IC50 = 8 nM T92072 CVR5X8 9974009 Ki = 42 nM T92072 CZE6O5 9975036 Ki = 4.4 nM T92072 CZVI16 9976651 EC50 = 501187233.6 nM T92072 COWM79 9977467 Ki = 100 nM T92072 C5SZL7 9978117 Ki = 0.44 nM T92072 CE1MT0 9978226 Ki = 100 nM T92072 CZ84DN 9981250 IC50 = 2000 nM T92072 CLI90J 9981945 Ki = 2450 nM T92072 CLZ2G0 9982930 Ki = 2230 nM T92072 C5F1IV 9985321 Ki = 325 nM T92072 C06EVM 9995603 Ki = 34 nM T92072 CJ83TP 9999033 Ki > 100000 nM T92072 CMP5T0 10007115 Ki = 710 nM T92072 C2WSC5 10014953 Ki > 10000 nM T92072 CAT43U 10016584 EC50 = 640 nM T92072 CPAT84 10020580 Ki = 18 nM T92072 CM3OS9 10021401 EC50 = 1.995 nM T92072 CD52TK 10022380 IC50 = 90 nM T92072 C2CQ8U 10022943 Ki = 125.89 nM T92072 C7KIA0 10023011 IC50 = 11000 nM T92072 CA4X5Z 10026670 Ki = 123 nM T92072 CU2YA5 10026817 IC50 = 14000 nM T92072 C0T4JM 10027485 IC50 = 700 nM T92072 CWUJ27 10028379 Ki = 630 nM T92072 C9E4GW 10029879 Ki > 6000 nM T92072 C5PF2I 10038941 Ki = 1.1 nM T92072 CP2ZS6 10039961 Ki > 10000 nM T92072 CJZY04 10040075 Ki = 168 nM T92072 CKD5L0 10043187 Ki = 0.3981 nM T92072 CX32QD 10046002 Ki = 20 nM T92072 CLRM29 10046145 Ki = 2500 nM T92072 CU7EA4 10047690 Ki = 34 nM T92072 C4H9QD 10048706 IC50 = 4200 nM T92072 C3X1QT 10050031 Ki = 432 nM T92072 C9JNZ4 10051921 IC50 = 60 nM T92072 C9SM7V 10052252 Ki > 6000 nM T92072 CX59SD 10062568 Ki = 124.7 nM T92072 C7EKU9 10063737 Ki = 70 nM T92072 CGE17I 10065148 Ki = 9 nM T92072 C0HBO3 10067267 Ki = 1 nM T92072 CCS38I 10067676 IC50 = 6300 nM T92072 CG56KA 10074917 IC50 = 20 nM T92072 C6VLS0 10075248 Ki = 122 nM T92072 C1W0YH 10083550 Ki = 1926 nM T92072 CSF1K3 10085767 Ki = 1460 nM T92072 CZ7JH1 10086671 EC50 = 1600 nM T92072 CFDU07 10090006 Ki = 1000 nM T92072 CEZ13D 10091878 IC50 = 7000 nM T92072 CKR13A 10094488 Ki = 125.89 nM T92072 C42KUZ 10108084 Ki = 2740 nM T92072 CAZJ75 10118562 Ki = 1361 nM T92072 CRTI50 10125973 EC50 = 50000 nM T92072 CFI6P8 10126989 Ki = 110 nM T92072 C78NYU 10131882 IC50 > 6200 nM T92072 C5WDR4 10132256 Ki = 560 nM T92072 CIN47Q 10132473 Ki = 624 nM T92072 C5JC6Y 10132529 Ki = 534 nM T92072 C1AU0B 10150517 Ki = 4200 nM T92072 CV87WF 10153029 IC50 = 59 nM T92072 CZ17TE 10153190 Ki > 1000 nM T92072 C6IC0Y 10154604 Ki = 1530 nM T92072 CBY63V 10155413 Ki = 100 nM T92072 C7OC0T 10156654 IC50 > 10000 nM T92072 C7J5EN 10158974 Ki > 6000 nM T92072 CRVU75 10164201 Ki > 6000 nM T92072 C4FNY6 10175278 Ki > 1000 nM T92072 CB39ZH 10179175 IC50 = 19.05 nM T92072 CUC8Y6 10196060 IC50 = 152 nM T92072 C5NOP9 10196114 Ki > 200 nM T92072 C1NW4L 10196517 IC50 = 205 nM T92072 CRY0O1 10200261 EC50 = 158489.32 nM T92072 C9KP1Y 10218183 IC50 = 102 nM T92072 CN9W0F 10225178 Ki = 8.1 nM T92072 CUH18Y 10236771 EC50 = 4200 nM T92072 C6A8EB 10237267 Ki = 66 nM T92072 C84YAW 10237847 IC50 = 68 nM T92072 CZE01H 10238677 IC50 = 123 nM T92072 CP7K3D 10246959 Ki = 1 nM T92072 C5RKX3 10247091 Ki > 100000 nM T92072 C2HVY5 10248379 Ki = 391 nM T92072 CH7VN4 10249674 Ki = 576 nM T92072 C0TXB5 10250190 Ki > 100000 nM T92072 C0CG8M 10253877 Ki = 2600 nM T92072 CGMN21 10254700 Ki = 7.4 nM T92072 CT41UJ 10256007 Ki = 670 nM T92072 C9RSB2 10256116 Ki = 700 nM T92072 CS80UL 10257979 Ki = 3548.13 nM T92072 C86SHK 10264202 Ki = 1.585 nM T92072 CF1UN5 10267860 Ki = 738 nM T92072 CN40IZ 10269215 Ki = 76 nM T92072 CWQ12V 10269216 Ki = 26 nM T92072 CYCI04 10269418 Ki = 70 nM T92072 CA1U9H 10269806 Ki = 3288 nM T92072 C2CQK6 10270416 Ki = 26 nM T92072 CF05LR 10275609 Ki = 50.12 nM T92072 C3MG6S 10278807 Ki = 602 nM T92072 C59HGD 10287615 EC50 = 17000 nM T92072 CVND46 10287779 Ki = 358 nM T92072 CB5DN6 10288169 IC50 = 150 nM T92072 CH6ZC0 10288197 IC50 = 54 nM T92072 CIQ18W 10291002 Ki = 28 nM T92072 CI5LZ3 10291235 Ki = 46 nM T92072 C8ZVR9 10291405 Ki = 231 nM T92072 C0VY4L 10291948 Ki = 197 nM T92072 C8RM9P 10292899 EC50 = 63095734.45 nM T92072 C40WZO 10296638 Ki = 7.6 nM T92072 CI2E8K 10308937 Ki = 1600 nM T92072 CU17KP 10310578 IC50 = 396 nM T92072 C8BO9X 10310768 Ki > 6000 nM T92072 CC21BD 10311222 IC50 = 415 nM T92072 CBSE14 10311510 Ki = 9 nM T92072 C0H5MU 10316176 Ki = 74.8 nM T92072 CXY40F 10318983 Ki = 179 nM T92072 C62MZJ 10320122 Ki = 10000 nM T92072 CJ8P0A 10320760 EC50 = 12500 nM T92072 CG6FS9 10320870 IC50 = 3500 nM T92072 C0SK5W 10322498 Ki = 419 nM T92072 C1S7MG 10342391 EC50 = 6360 nM T92072 CZ81IA 10342970 Ki = 766 nM T92072 C0XHI4 10345159 Ki = 20.7 nM T92072 C7IPE9 10346511 Ki = 17 nM T92072 CF4UB5 10357057 Ki = 1700 nM T92072 CD7C2A 10359522 Ki = 50 nM T92072 C1RFV6 10362099 Ki = 253 nM T92072 CKJE75 10366048 IC50 = 1200 nM T92072 C04LWE 10367224 IC50 = 700 nM T92072 CFT42V 10368871 IC50 = 21 nM T92072 CAL97Z 10368912 IC50 = 80 nM T92072 C2R9YK 10369458 Ki = 12100 nM T92072 CHZ32J 10377463 Ki = 5.623 nM T92072 C5FLB1 10386251 IC50 = 4000 nM T92072 CM8TS4 10387069 IC50 = 600 nM T92072 C5HPZ3 10387088 Ki = 149 nM T92072 CUP34N 10388920 Ki = 50 nM T92072 CLW3V4 10390375 IC50 = 800 nM T92072 CPF60T 10391480 IC50 = 87 nM T92072 C5F4WP 10403711 Ki = 1.9 nM T92072 C4UX5I 10404217 Ki = 1181 nM T92072 CN6TD0 10405277 IC50 > 100000 nM T92072 C3GYR7 10411021 IC50 = 11 nM T92072 C47SOT 10413798 IC50 = 8.7 nM T92072 CAJ68I 10426659 Ki = 3420 nM T92072 CWUB34 10431614 Ki = 430 nM T92072 CMX8S3 10435244 IC50 = 2600 nM T92072 CO4H0C 10436433 Ki > 10000 nM T92072 CP4XJ5 10445452 Ki = 0.4 nM T92072 C6BH4D 10449090 Ki = 3.29 nM T92072 CSD86M 10449535 Ki = 5.5 nM T92072 C8XFL5 10449783 Ki = 19.95 nM T92072 CZ9VB4 10450691 Ki = 2100 nM T92072 C1BW6K 10451086 Ki = 1.259 nM T92072 C9OXR2 10451887 IC50 = 17000 nM T92072 C9FQ6C 10452788 Ki = 68 nM T92072 CK9FA7 10453097 Ki = 700 nM T92072 C0BYA5 10453675 IC50 = 2200 nM T92072 CM4C2X 10455080 Ki = 3.4 nM T92072 CGM46Y 10455852 Ki = 1.7 nM T92072 C8MP2K 10455955 IC50 = 20 nM T92072 C4OMF3 10468228 Ki = 2 nM T92072 C2KJO9 10469918 EC50 = 2400 nM T92072 C15VAO 10471588 Ki = 36 nM T92072 CKL5T7 10481731 IC50 = 16.8 nM T92072 C93CAI 10494738 Ki > 10000 nM T92072 CHC23X 10505816 Ki = 251 nM T92072 CCP12B 10537885 Ki > 10000 nM T92072 CJ8H1E 10538858 Ki = 490 nM T92072 CFOS68 10539663 Ki = 211 nM T92072 CQIC13 10539682 Ki = 1258.93 nM T92072 CLD25R 10540853 Ki = 79.43 nM T92072 C5ATC3 10541585 Ki = 19.95 nM T92072 CA2BP3 10544916 Ki = 25 nM T92072 C2K6RI 10562783 Ki = 2000 nM T92072 CL23DC 10580789 Ki = 255 nM T92072 CEW4T3 10587109 Ki = 101 nM T92072 C02GZY 10601859 Ki = 1500 nM T92072 CS2VT6 10605011 Ki = 389 nM T92072 C6M1NH 10613770 Ki = 31.62 nM T92072 C2N5UX 10616023 Ki = 30 nM T92072 CJ06HI 10618828 Ki = 19 nM T92072 CGMH35 10619822 Ki = 87.8 nM T92072 C8JB3I 10623248 Ki = 296 nM T92072 CY6QP1 10626463 Ki = 3164 nM T92072 C7QWO6 10637742 Ki = 14 nM T92072 C78YHS 10641040 Ki = 1000 nM T92072 C7LN3U 10642208 Ki = 1.585 nM T92072 C8O4LD 10645750 Ki = 1650 nM T92072 C8O2UT 10647227 Ki = 245 nM T92072 CBI7X5 10659581 Ki = 5 nM T92072 CZ97XY 10661229 Ki = 176.4 nM T92072 C8NCG3 10661707 Ki = 175 nM T92072 CKG51X 10663067 Ki = 25.12 nM T92072 C0U2LA 10665761 Ki = 29 nM T92072 CVIR83 10667072 Ki = 3.981 nM T92072 CHQ6B9 10668865 Ki = 2170 nM T92072 CR2MJ6 10687275 Ki = 1995.26 nM T92072 CGU6W0 10687707 Ki = 316.23 nM T92072 CWJ60V 10691124 Ki = 27 nM T92072 C9B1PF 10696675 Ki = 251 nM T92072 CLZ7M1 10706862 Ki = 5.012 nM T92072 C5EM0D 10709852 Ki = 69 nM T92072 C4PXZ8 10712345 Ki = 981 nM T92072 C07JSG 10720065 Ki = 49.7 nM T92072 CKIR94 10728732 Ki = 1400 nM T92072 CJ8Z2O 10729354 Ki = 6309.57 nM T92072 CKMJ53 10732242 Ki = 40 nM T92072 C9IJL3 10734376 Ki = 2000 nM T92072 C7NXS3 10737168 Ki = 3 nM T92072 C9DP7L 10744124 IC50 = 101 nM T92072 CB0L1T 10745111 Ki = 2466 nM T92072 C03CBY 10755990 Ki = 19.95 nM T92072 CSZW84 10757861 Ki = 31.62 nM T92072 CWK2M9 10761106 Ki = 15 nM T92072 CUG21I 10761800 Ki = 130 nM T92072 C5D8YL 10763173 Ki = 79.43 nM T92072 CCZ4U8 10765059 Ki = 1531 nM T92072 C34RFS 10765882 IC50 = 165 nM T92072 CY3H0T 10766957 IC50 = 112 nM T92072 CK0C8P 10767043 Ki = 17.9 nM T92072 C5B6KP 10769581 Ki = 247 nM T92072 CB9I0J 10778032 Ki = 501.19 nM T92072 CIRS48 10778887 Ki = 10 nM T92072 C3GJ5Z 10779327 Ki = 10 nM T92072 CNC32V 10785815 Ki = 5.012 nM T92072 C79MNZ 10791347 Ki = 201 nM T92072 CYG2J5 10792296 Ki = 61.2 nM T92072 CNX03D 10798671 Ki = 10000 nM T92072 C7U4RN 10801510 Ki > 10000 nM T92072 C7BT0O 10824674 Ki = 25 nM T92072 CQ01KP 10824688 Ki = 5011.87 nM T92072 C1TP5N 10828916 Ki = 794.33 nM T92072 C6UP5K 10834513 Ki = 348 nM T92072 C2E6PX 10839228 Ki = 105 nM T92072 C20WTU 10839296 Ki = 57 nM T92072 C1TS0R 10839674 IC50 = 24.9 nM T92072 C89OKC 10840167 Ki = 73.5 nM T92072 C6GIK9 10847356 Ki = 15.85 nM T92072 C6CSZ4 10852375 Ki = 5.42 nM T92072 CE04SL 10852506 Ki = 2 nM T92072 C3I2WZ 10859484 Ki = 50 nM T92072 C3QWZ1 10862463 Ki = 429 nM T92072 CZ7WJ9 10863425 Ki = 526 nM T92072 C4J8CR 10868826 Ki = 2400 nM T92072 C7RD3K 10872091 Ki > 10000 nM T92072 C4HO6X 10874051 Ki = 70 nM T92072 C1AL7H 10884000 Ki = 175 nM T92072 CN8J0Y 10884265 Ki = 1015 nM T92072 CY62BK 10884803 Ki = 1214 nM T92072 C9YZ3M 10885937 Ki = 68 nM T92072 CIG9Z2 10895416 Ki = 325 nM T92072 C2P1QB 10895565 Ki = 55 nM T92072 C2LV6K 10904370 Ki = 235 nM T92072 CU93CT 10904839 Ki = 2160 nM T92072 C3KOX6 10905184 Ki = 731 nM T92072 CKV30L 10905799 Ki = 409 nM T92072 CH52LS 10906943 Ki = 142 nM T92072 C4H8PS 10914466 Ki = 350 nM T92072 CI87AW 10915653 Ki = 43 nM T92072 CJ52TM 10916451 Ki = 4927 nM T92072 CS58FH 10917575 Ki = 70 nM T92072 CWU29C 10917670 Ki = 773 nM T92072 CVFL61 10918042 Ki = 300 nM T92072 CQXA29 10926253 Ki = 30 nM T92072 CJB64E 10927693 Ki = 400 nM T92072 CFZ49H 10928011 Ki = 2630 nM T92072 C1B6XL 10928182 Ki = 250 nM T92072 CG2N7W 10928649 Ki = 584 nM T92072 C58CRE 10938276 Ki = 262 nM T92072 CG24MW 10938325 Ki = 1026 nM T92072 C6FQ3L 10938608 Ki = 302 nM T92072 C8BLN4 10939224 Ki = 842 nM T92072 CXWV50 10959335 Ki = 75 nM T92072 CY2OS9 10961304 Ki = 150 nM T92072 C7YVC5 10962009 Ki = 9399 nM T92072 CKE84F 10970819 Ki = 138 nM T92072 CD16UB 10971099 Ki = 714 nM T92072 C9WLT0 10971427 Ki = 419 nM T92072 C6OFK0 10971806 Ki = 400 nM T92072 C4ZU8F 10971841 Ki = 376 nM T92072 CBW9J6 10972594 Ki = 4965 nM T92072 C4G0YQ 10982985 Ki = 300 nM T92072 C83XMH 10993869 Ki = 139 nM T92072 C6BH4T 10993916 Ki = 750 nM T92072 C9NP1R 10994142 Ki > 1000 nM T92072 C3F4TJ 10994183 Ki = 410 nM T92072 CSO19C 10994216 Ki = 120 nM T92072 C31HJV 10994317 Ki = 400 nM T92072 CJ6C9K 11003971 IC50 = 344 nM T92072 CMDB43 11004373 Ki = 348 nM T92072 CEP35L 11004986 Ki > 1000 nM T92072 CLR4B8 11005067 Ki = 558 nM T92072 C69NZT 11005362 Ki = 443 nM T92072 C2SNI1 11005491 Ki = 579 nM T92072 C2QJW7 11013957 Ki = 83 nM T92072 C0KDE3 11014188 Ki = 702 nM T92072 C47IDH 11014608 Ki = 43 nM T92072 C6EQD3 11015003 Ki = 602 nM T92072 C5BQ0H 11015572 Ki = 1700 nM T92072 C30WTZ 11017082 Ki = 5297 nM T92072 CI3E7D 11019436 Ki > 100000 nM T92072 C8UPZ3 11026001 Ki = 9.6 nM T92072 CF5B8Z 11026358 Ki > 1000 nM T92072 CPD61T 11026434 Ki = 1134 nM T92072 C12YXH 11027282 Ki = 6392 nM T92072 CX28EA 11027412 Ki = 50 nM T92072 CPV27K 11027743 Ki = 12100 nM T92072 CW05DS 11028588 Ki > 1000 nM T92072 C5I8UZ 11035880 Ki = 179 nM T92072 CHEA89 11037671 Ki = 4197 nM T92072 CR7FM2 11037739 Ki = 300 nM T92072 CM9FK6 11037972 Ki = 500 nM T92072 CUV0P9 11046285 Ki = 28 nM T92072 CS8P0U 11048163 Ki = 190 nM T92072 CL1RP8 11048438 Ki = 1.1 nM T92072 CW7Q6U 11053743 Ki = 31 nM T92072 CL29NE 11056301 Ki = 325 nM T92072 CCS8A6 11058550 Ki = 450 nM T92072 CFJG64 11059058 IC50 = 2640 nM T92072 CYZ83I 11059351 Ki = 200 nM T92072 CA91IB 11060260 Ki = 369 nM T92072 CM7TR4 11068963 Ki = 1690 nM T92072 C9KRQ1 11070905 Ki > 10000 nM T92072 C7HIP2 11071159 Ki = 316 nM T92072 CN5S7E 11078951 Ki = 666 nM T92072 C1EJI0 11080491 Ki = 200 nM T92072 CKX4G6 11080788 Ki = 248 nM T92072 C4Y7NZ 11081189 Ki = 611 nM T92072 C83TJN 11090423 Ki = 1460 nM T92072 CR3X1M 11091600 Ki = 80 nM T92072 C64PWO 11091632 Ki = 280 nM T92072 C15EQZ 11091783 Ki = 136 nM T92072 CZW34N 11099564 Ki = 124 nM T92072 CVDM13 11102838 Ki = 780 nM T92072 CMY97P 11112381 Ki = 7.1 nM T92072 C3Z5PU 11112543 Ki = 300 nM T92072 C6RB5D 11112711 Ki = 2.2 nM T92072 C3IFX4 11112849 Ki = 802 nM T92072 CR7X2T 11122708 Ki = 400 nM T92072 CLN23H 11123135 Ki > 1000 nM T92072 C06JLD 11123887 Ki > 10000 nM T92072 C4CWA8 11133107 Ki > 1000 nM T92072 CJ86ZM 11133545 Ki = 1115 nM T92072 CL19OW 11133804 Ki = 275 nM T92072 CTG5Y7 11133843 Ki = 318 nM T92072 CH4TG2 11144119 Ki > 1000 nM T92072 C9N1RL 11144868 Ki = 600 nM T92072 C72QCG 11145314 Ki = 9330 nM T92072 C4AR0D 11150120 Ki = 339.5 nM T92072 CVF8Z5 11151115 Ki > 10000 nM T92072 C79YSE 11153187 Ki > 1000 nM T92072 CM9SW5 11154129 Ki = 220 nM T92072 CLQR16 11157262 Ki = 310 nM T92072 C1FVD5 11162618 Ki = 38 nM T92072 CNY65E 11163483 Ki = 320 nM T92072 CJ0T6F 11163971 Ki = 210 nM T92072 CS0N2C 11164346 Ki = 7 nM T92072 CPB62L 11174953 Ki = 2.4 nM T92072 C12UTW 11175566 Ki > 1000 nM T92072 CFL0O8 11177363 Ki = 1510 nM T92072 CJ02LB 11178828 Ki = 3700 nM T92072 CGKV50 11186097 Ki = 39.81 nM T92072 CHD65Q 11198201 Ki = 65 nM T92072 C0L4GE 11199718 Ki = 1995.26 nM T92072 CD7QP2 11199731 Ki = 978 nM T92072 CS6D8T 11200454 Ki = 6309.57 nM T92072 C41PYH 11209919 Ki > 1000 nM T92072 C6JD3L 11210192 Ki = 108.9 nM T92072 CV5Y6A 11214123 Ki = 881 nM T92072 CUNM43 11220580 Ki = 97 nM T92072 CH28VP 11221189 Ki = 107 nM T92072 C3FP0D 11229946 Ki = 24 nM T92072 CK5P7G 11232232 Ki = 299 nM T92072 C3B4ZF 11232994 Ki = 1940 nM T92072 C9IHT1 11233411 Ki > 1000 nM T92072 CB6Y4A 11233413 Ki > 1000 nM T92072 C57WSV 11244376 Ki = 6.49 nM T92072 CES2X9 11255221 Ki > 10000 nM T92072 CA4EP9 11255271 Ki = 1070.5 nM T92072 CPZ8A2 11255409 Ki = 12 nM T92072 COYW84 11255849 Ki = 41 nM T92072 C7LS3R 11256992 Ki = 2 nM T92072 CCU71Z 11257069 Ki > 1000 nM T92072 C86XNQ 11260448 Ki = 740 nM T92072 CH0U1C 11266371 Ki = 930 nM T92072 CK7SM8 11266431 Ki = 592.8 nM T92072 CR7C8S 11268516 Ki = 150 nM T92072 CDL7O5 11277831 Ki > 10000 nM T92072 CYWN16 11278445 Ki = 430 nM T92072 C45RAF 11289724 Ki = 7500 nM T92072 CGR1A8 11289861 Ki = 131 nM T92072 C48JAP 11290020 Ki = 24.9 nM T92072 C8B2RV 11290216 Ki = 186 nM T92072 C8A0MT 11290634 Ki = 1086 nM T92072 C46LIX 11301348 Ki = 49 nM T92072 CLW5H2 11301432 Ki = 960 nM T92072 C3Y1OW 11302050 Ki = 1208 nM T92072 CQ7O1I 11302588 Ki = 3900 nM T92072 C4PH8A 11306173 Ki = 910 nM T92072 CJ4MT0 11311283 Ki = 6.31 nM T92072 CDC83I 11312454 Ki = 1342 nM T92072 CX09ZQ 11312833 Ki > 10000 nM T92072 CGB03H 11313388 Ki = 463 nM T92072 CCMS25 11313542 Ki = 1100 nM T92072 CO1Q4Y 11313543 Ki = 460 nM T92072 CUS2N9 11313850 Ki > 1000 nM T92072 C67CZB 11314995 Ki = 30 nM T92072 CX7QW0 11324734 Ki = 1880 nM T92072 C5UMJ9 11324754 Ki = 151 nM T92072 CY8KX5 11329375 Ki = 240 nM T92072 CJX89P 11348709 Ki > 1000 nM T92072 CEU9X7 11348760 Ki > 10000 nM T92072 C1Q8NA 11348867 Ki = 15.5 nM T92072 C3TH4B 11352497 Ki = 600 nM T92072 C1C2NM 11359310 Ki = 4.3 nM T92072 CK7M5J 11359476 Ki = 224 nM T92072 CRND96 11360082 Ki > 1000 nM T92072 CT8J7Q 11368737 Ki = 25.12 nM T92072 C1WQU8 11369938 Ki = 15 nM T92072 C8G3FO 11371101 Ki > 1000 nM T92072 CB8RU3 11380183 Ki = 9.2 nM T92072 C0M8KH 11380777 Ki = 4400.5 nM T92072 CB3J6T 11380878 Ki = 124 nM T92072 CRU3A7 11381738 Ki = 47 nM T92072 C3IHK7 11381773 Ki = 166 nM T92072 CR73JH 11382077 Ki = 650 nM T92072 CSD31L 11386134 Ki = 10000 nM T92072 C8KD6J 11386951 Ki > 10000 nM T92072 CJ9WG8 11391873 Ki = 2200 nM T92072 CK58UE 11391964 Ki = 214 nM T92072 CB2C4P 11392671 Ki = 73 nM T92072 C0A6MY 11392863 Ki = 81 nM T92072 CVAJ46 11393155 Ki = 34.5 nM T92072 CXPM05 11394389 Ki = 350 nM T92072 C1CL4W 11404060 Ki = 4212 nM T92072 C6IVY0 11408692 Ki = 1.63 nM T92072 CLM04X 11412911 Ki > 10000 nM T92072 CD9PL7 11415171 Ki = 316.23 nM T92072 C3NO7I 11415926 Ki = 79.43 nM T92072 CS7ZX2 11416448 Ki = 1401 nM T92072 CCW60O 11420226 Ki = 200 nM T92072 CDVM74 11424338 Ki > 10000 nM T92072 C30ZXP 11426423 Ki = 122 nM T92072 CQ7H6Z 11427378 Ki = 890.3 nM T92072 CPF8K7 11427490 Ki = 504 nM T92072 CPS9L6 11427880 Ki = 2.14 nM T92072 CSJ2X5 11428282 Ki = 119 nM T92072 CF4H1A 11428535 Ki = 460 nM T92072 C85LYP 11430418 IC50 > 1000 nM T92072 C1U0CT 11431149 Ki = 20.6 nM T92072 CF8EN7 11437060 Ki = 10000 nM T92072 CF2PT3 11449747 Ki = 81 nM T92072 C7D3AN 11451298 Ki = 39.81 nM T92072 C6CV1B 11452333 Ki > 1000 nM T92072 CA6YD2 11461202 Ki = 7.58 nM T92072 CZIN71 11462033 Ki = 2.14 nM T92072 C35UFZ 11462655 Ki = 14 nM T92072 C5M3SD 11463674 Ki > 1000 nM T92072 C5JTD0 11464552 Ki > 1000 nM T92072 CUP24K 11464737 EC50 = 11600 nM T92072 C9CFK5 11465677 Ki > 1000 nM T92072 C9NP2C 11466670 Ki = 2300 nM T92072 CDY79C 11472819 Ki = 260 nM T92072 CFN40B 11473008 Ki = 27.7 nM T92072 CK9VD0 11473488 Ki = 1100 nM T92072 C9RK6X 11475577 Ki > 1000 nM T92072 C83XMS 11475769 Ki = 3800 nM T92072 CE7JS1 11483771 Ki = 54 nM T92072 C2SY3I 11492651 Ki > 100000 nM T92072 CI4JC0 11492857 Ki = 3.2 nM T92072 CL49IS 11493754 Ki > 6000 nM T92072 CKN80I 11494063 Ki = 373 nM T92072 C5FY2G 11494318 Ki = 1056.3 nM T92072 CTM2U8 11494728 Ki = 3981.07 nM T92072 CZ0FN7 11494993 Ki = 31.62 nM T92072 CO32QT 11495161 Ki = 22 nM T92072 CH7UC9 11495611 Ki = 59 nM T92072 C5LN1D 11497238 Ki = 330 nM T92072 C3YG6W 11500266 Ki = 2.1 nM T92072 C6KL3S 11501678 Ki = 210 nM T92072 CD0T6O 11503200 Ki = 530 nM T92072 C0WV8M 11507345 Ki > 10000 nM T92072 COG79X 11508049 Ki = 10 nM T92072 C0AWD8 11508923 Ki = 350 nM T92072 C8GL1J 11511804 Ki > 1000 nM T92072 CYN5U6 11511897 Ki = 2190 nM T92072 CH03ZF 11516748 Ki > 1000 nM T92072 CN2DI8 11516857 Ki = 638 nM T92072 CD29AZ 11517013 Ki > 1000 nM T92072 C81KTQ 11518657 Ki = 199.53 nM T92072 CT60SW 11522152 Ki = 11500 nM T92072 CQNA38 11522379 Ki = 2.86 nM T92072 CS1M7B 11522670 Ki = 75 nM T92072 CQZ37L 11524264 Ki > 1000 nM T92072 CH9DU2 11524593 Ki = 1400 nM T92072 C23LEU 11524637 Ki = 34 nM T92072 C1CJ2S 11525283 Ki = 183 nM T92072 C5BVY4 11525912 Ki = 19.95 nM T92072 CVR6D0 11527363 EC50 = 1 nM T92072 C21IUQ 11529194 Ki > 10000 nM T92072 CKC6F5 11529450 Ki = 6 nM T92072 CV2DP6 11530256 Ki = 3850 nM T92072 C6Z0EX 11531100 Ki = 3.7 nM T92072 C46UMB 11531355 Ki = 98 nM T92072 C1M4HF 11531697 Ki = 199.53 nM T92072 CEDZ81 11532717 Ki = 190 nM T92072 C6HAF9 11533237 Ki = 3100 nM T92072 C92FYA 11533614 EC50 > 10000 nM T92072 CYWJ05 11535816 Ki > 10000 nM T92072 C8P2YI 11536894 Ki = 6.2 nM T92072 C0Z9UA 11536947 Ki = 9.3 nM T92072 CU38FS 11537425 Ki > 10000 nM T92072 CH43JG 11538373 Ki > 1000 nM T92072 C5KDX9 11539152 Ki > 30000 nM T92072 C16FKE 11544506 Ki > 10000 nM T92072 CT6C5U 11544894 Ki = 460 nM T92072 CW62MV 11545273 Ki = 230 nM T92072 C2QHP4 11545341 Ki = 770 nM T92072 CNOW78 11546087 Ki = 1000 nM T92072 CPNA09 11546129 Ki = 1000 nM T92072 CUD5B0 11546358 Ki > 1000 nM T92072 CRCP28 11546394 Ki = 1995.26 nM T92072 C1U8RO 11547107 Ki = 41 nM T92072 CPV7Y8 11553016 Ki > 10000 nM T92072 C3IET8 11553509 Ki = 7.762 nM T92072 C6CVK7 11555032 Ki > 1000 nM T92072 C7A9PY 11557440 Ki > 10000 nM T92072 C0VES1 11560202 Ki = 550 nM T92072 C7VD3G 11560510 Ki = 48 nM T92072 C7T4KL 11561727 Ki = 19.95 nM T92072 C49FXT 11562106 Ki = 79.43 nM T92072 C41AXZ 11565780 Ki = 15 nM T92072 CIR70L 11565927 Ki > 10000 nM T92072 C93ANH 11568001 Ki = 14.79 nM T92072 C9WVP1 11568203 Ki = 441 nM T92072 C85MGW 11568359 Ki = 185 nM T92072 CLV6H3 11568586 Ki = 507 nM T92072 C37CAT 11569026 Ki = 430 nM T92072 CY3C0A 11573708 Ki = 82 nM T92072 C9VP0G 11574573 EC50 > 10000 nM T92072 CZIP72 11574851 Ki = 158.49 nM T92072 CGY1A2 11575180 Ki = 1000 nM T92072 CQTN95 11575377 Ki = 125.89 nM T92072 C7RA2X 11575498 Ki = 31 nM T92072 CVQ19R 11577804 Ki = 144 nM T92072 CZ65AS 11580284 Ki = 370 nM T92072 C5JOW8 11580374 Ki = 5.7 nM T92072 C8Y9LA 11582537 Ki = 620 nM T92072 CAR2U3 11582578 Ki = 59 nM T92072 C5I4RZ 11582697 Ki = 7 nM T92072 CYP80S 11582743 Ki = 1995.26 nM T92072 CWF57T 11583760 Ki = 50.12 nM T92072 C6D1MA 11584660 Ki > 15848.93 nM T92072 CN62XG 11585280 IC50 = 760 nM T92072 CTG7A1 11585567 Ki = 1710 nM T92072 C0TFK3 11586663 Ki = 340 nM T92072 CM62BJ 11587409 Ki = 2.8 nM T92072 CYJ29E 11587927 Ki = 6.5 nM T92072 C8S2RC 11588630 Ki = 580 nM T92072 CN7T8C 11589094 Ki = 47.8 nM T92072 CU0MX8 11589625 Ki = 19 nM T92072 CS1RK4 11595040 Ki > 30000 nM T92072 CNTA30 11595292 Ki = 210 nM T92072 C1ERP7 11595710 Ki = 2700 nM T92072 CGPE63 11596214 Ki = 2100 nM T92072 CUXN24 11596614 Ki = 38 nM T92072 C31YOR 11596733 Ki = 265 nM T92072 C8OJ6R 11597583 Ki = 1600 nM T92072 CQIT47 11598485 Ki = 39.81 nM T92072 CC72QD 11598486 Ki = 100 nM T92072 CVN1Y5 11601342 Ki > 10000 nM T92072 C1QJ4W 11602451 Ki = 27 nM T92072 C80ZIV 11602914 Ki = 4170 nM T92072 CYHI46 11603727 Ki = 10000 nM T92072 CAC54T 11606834 Ki = 126 nM T92072 C21IGF 11608581 Ki = 266 nM T92072 CB06AO 11608818 Ki > 100000 nM T92072 C8LA0I 11609235 Ki = 55 nM T92072 CPS1A9 11609536 Ki = 41 nM T92072 CWMD07 11610638 Ki = 380 nM T92072 CA5B6V 11611370 Ki = 4070 nM T92072 C6NID5 11611580 Ki = 390 nM T92072 CXB6L3 11611815 Ki = 79.43 nM T92072 C42QLP 11611903 Ki > 10000 nM T92072 C2G4JX 11612320 Ki = 44 nM T92072 CC8Q7O 11612367 Ki = 31.62 nM T92072 CKH3X2 11618263 Ki = 19.95 nM T92072 CVW0B6 11618482 Ki = 3162.28 nM T92072 C39ZVR 11618633 Ki = 77 nM T92072 CVN84J 11618812 Ki = 1995.26 nM T92072 CF09KT 11619671 Ki = 558 nM T92072 CSX24T 11619688 Ki = 31.62 nM T92072 CLV26W 11623708 Ki = 3.9 nM T92072 C7AM8B 11623934 Ki = 10 nM T92072 CVL8P5 11625174 Ki = 37.3 nM T92072 CJDZ72 11625255 Ki = 25 nM T92072 C2OD7U 11625772 Ki = 13.9 nM T92072 C35XDW 11625796 Ki > 1000 nM T92072 CDM6N2 11626876 Ki = 12.59 nM T92072 C02QTY 11630237 Ki = 496 nM T92072 C0JOM4 11630922 Ki > 30000 nM T92072 C57HNQ 11631512 Ki = 27 nM T92072 CXSZ13 11632013 Ki = 650 nM T92072 CJ5OM1 11632785 Ki = 239.88 nM T92072 CJ02TL 11633189 Ki = 70 nM T92072 C9JO8B 11633747 Ki = 1258.93 nM T92072 C7TFE5 11634270 Ki = 76.7 nM T92072 CX2B4O 11638430 Ki = 150 nM T92072 CFTH84 11638790 Ki > 10000 nM T92072 CH0K6M 11639132 Ki = 180 nM T92072 C42QLC 11639150 Ki > 10000 nM T92072 C1LIP2 11640419 Ki = 37 nM T92072 CXUQ86 11640487 Ki = 2 nM T92072 C80FAW 11640539 Ki = 4.266 nM T92072 CG20LN 11640941 Ki = 15.85 nM T92072 CM39TC 11641365 Ki = 18.8 nM T92072 C85ZEB 11642035 Ki = 32.36 nM T92072 CEC6Z2 11646441 Ki = 158.49 nM T92072 C5BH2I 11647009 Ki = 158.49 nM T92072 C9X5JF 11647607 Ki = 170 nM T92072 C3VZF7 11649145 Ki = 10.96 nM T92072 CND50M 11649544 Ki = 21 nM T92072 CT6CW3 11650023 Ki = 92 nM T92072 CAX46N 11654460 Ki = 170 nM T92072 CIS7K1 11654461 Ki = 23 nM T92072 CC8X7R 11655061 Ki = 830 nM T92072 C60BFR 11656087 Ki = 63.1 nM T92072 CM54YT 11657274 Ki = 1720 nM T92072 CWY7T6 11659363 Ki = 8 nM T92072 C1JU7A 11659696 IC50 = 45 nM T92072 C1XYR3 11659733 Ki = 205 nM T92072 CX49RB 11662217 Ki = 10000 nM T92072 CU94XB 11662646 Ki = 75.8 nM T92072 CU8Q7J 11662647 Ki = 10000 nM T92072 C1R2UX 11662937 Ki = 63.1 nM T92072 CV39AR 11662965 EC50 > 10000 nM T92072 CQ13SY 11663152 Ki = 1980 nM T92072 CGA72F 11663932 Ki > 10000 nM T92072 CI2SK9 11667107 Ki > 10000 nM T92072 CGI6Y3 11667703 Ki > 1000 nM T92072 CB1Z8M 11667955 Ki = 340 nM T92072 C8SX1P 11667956 Ki = 260 nM T92072 CK3PZ9 11668813 Ki = 50.12 nM T92072 CEWR60 11670428 Ki = 7.943 nM T92072 CVPM67 11673316 Ki = 2270 nM T92072 CX95RT 11674018 Ki = 310 nM T92072 CZ6V5H 11675684 Ki = 3.2 nM T92072 CU90TV 11675940 Ki = 4.6 nM T92072 CV68PN 11676743 Ki = 630.96 nM T92072 C16PMS 11678491 Ki = 5870 nM T92072 C1I6FC 11680901 Ki = 242 nM T92072 CKU6E7 11681092 Ki = 6.2 nM T92072 CFD86C 11681113 Ki = 10 nM T92072 CF54VW 11681354 Ki = 25 nM T92072 CE8WD5 11681429 Ki = 18 nM T92072 CI8AX3 11683024 Ki = 245 nM T92072 CCSO04 11684389 Ki = 10 nM T92072 CAS80N 11684443 Ki = 18.2 nM T92072 CH30ES 11684672 Ki > 1000 nM T92072 CEU52V 11684979 Ki = 400 nM T92072 C4SWY5 11687423 Ki > 10000 nM T92072 CYFJ70 11687483 Ki = 101 nM T92072 CT3JM9 11690561 Ki = 570 nM T92072 CI10PQ 11690712 Ki = 54.8 nM T92072 C30UZA 11691773 Ki = 39.81 nM T92072 CZE9A8 11698568 Ki = 50.12 nM T92072 CH6Q2D 11698898 Ki = 2900 nM T92072 C2V3PS 11699353 EC50 > 10000 nM T92072 CWA0C8 11701717 Ki = 966 nM T92072 C69PJB 11702501 Ki = 80 nM T92072 C6HFY9 11703084 Ki = 270 nM T92072 C4RSG1 11703434 Ki = 251.19 nM T92072 CZ9IX2 11703893 Ki > 1000 nM T92072 CZE9V5 11705261 Ki = 370 nM T92072 C7BH9E 11705321 Ki = 125.89 nM T92072 CR6A2V 11709311 Ki = 8 nM T92072 CX6E5A 11709650 Ki = 37 nM T92072 C2LMK1 11711190 Ki = 17 nM T92072 CW0A6R 11711313 Ki = 100 nM T92072 CYI8O4 11711438 Ki = 350 nM T92072 CY48OK 11715751 Ki > 10000 nM T92072 CUM0C9 11716303 Ki = 3.6 nM T92072 CNR71Y 11717537 Ki > 1000 nM T92072 CD72OJ 11717832 Ki = 476 nM T92072 CYO9A7 11719640 Ki = 6.31 nM T92072 C6BEA8 11719675 Ki = 15.85 nM T92072 CH5DB1 11720501 Ki > 1000 nM T92072 C5P4YO 11723628 Ki = 870 nM T92072 C9J4WY 11728711 Ki = 6496 nM T92072 CAMT16 11728808 Ki = 326 nM T92072 CNT64M 11729275 Ki > 10000 nM T92072 CR80CF 11731871 Ki > 1000 nM T92072 C5GO4E 11732736 Ki = 281 nM T92072 CHW0A6 11733496 Ki = 75 nM T92072 CG7Y4O 11733556 Ki = 350 nM T92072 CF9Q7M 11733601 Ki = 350 nM T92072 CP2J9D 11738790 Ki = 1720 nM T92072 C43GFZ 11739282 Ki = 42 nM T92072 CNA2T5 11739287 Ki = 245 nM T92072 CLVT69 11739950 Ki = 34 nM T92072 C7OWV2 11740457 IC50 = 21 nM T92072 C0WNR6 11747281 Ki = 2100 nM T92072 CSR32T 11761221 Ki = 176 nM T92072 C7MD4U 11761823 Ki = 4494 nM T92072 CGSN15 11762418 Ki > 10000 nM T92072 CI82XE 11762982 Ki = 90 nM T92072 COFP43 11765357 IC50 = 3500 nM T92072 CE3D9A 11771825 Ki = 50.12 nM T92072 CMQ6D0 11773400 Ki = 156 nM T92072 CT84IV 11774108 Ki > 1000 nM T92072 CO76RZ 11782906 Ki = 89.2 nM T92072 CLPT97 11784369 Ki = 351 nM T92072 CBZJ16 11798195 Ki = 175 nM T92072 CV7T3H 11798368 Ki = 100 nM T92072 C8ZRL4 11801496 Ki = 293 nM T92072 CYN01G 11808994 Ki = 65 nM T92072 C1ZQF6 11811544 Ki = 500 nM T92072 CPMB38 11811761 Ki = 602 nM T92072 C82LEP 11812897 Ki = 708 nM T92072 C6ANG8 11813241 Ki = 2495 nM T92072 CZ52VY 11813713 Ki = 193 nM T92072 C4W2ID 11824950 Ki = 260 nM T92072 CP5A4S 11825841 Ki = 501.19 nM T92072 C31FGJ 11826577 Ki = 450 nM T92072 C15NOJ 11826924 Ki = 20 nM T92072 CAPF41 11850015 Ki = 104.3 nM T92072 CN54TL 11850295 IC50 = 5.1 nM T92072 CXLW54 11948707 Ki > 10000 nM T92072 C6Y3GI 11952504 Ki = 717 nM T92072 C3Y9JS 11952559 Ki = 2444 nM T92072 C9AVS8 11952560 Ki = 478 nM T92072 CD41JX 11952564 Ki = 82 nM T92072 CI6SX1 11952665 Ki = 252 nM T92072 C8OKX0 11952670 Ki = 357 nM T92072 CK3T8W 11953248 Ki = 317 nM T92072 CO29QE 11956192 Ki = 63 nM T92072 CM0SL3 11956193 Ki = 266 nM T92072 CW8KI0 11956198 Ki = 720 nM T92072 C6JVN1 11965767 Ki = 132 nM T92072 C0KXU5 11977965 Ki = 0.9 nM T92072 CXT4S5 11977966 Ki = 9 nM T92072 CWF2B7 11977967 Ki = 0.6 nM T92072 CULI10 11978309 Ki = 8 nM T92072 C6Z3SF 11978310 Ki = 30 nM T92072 C1EAC3 11978313 Ki = 2 nM T92072 CUVN07 11978421 Ki = 34 nM T92072 CPW02D 11995251 Ki = 59 nM T92072 C5YU6W 11995348 Ki = 171 nM T92072 C02DIG 11995349 Ki = 12 nM T92072 CTB21R 11995351 Ki = 109 nM T92072 CD25UB 11995352 Ki = 12 nM T92072 C1UGS4 11995353 Ki = 6 nM T92072 CE53IF 11995448 Ki = 22 nM T92072 C8TD1Y 11995554 Ki = 41 nM T92072 CI1TL9 11995555 Ki = 46 nM T92072 CUM6T1 11995557 Ki = 8 nM T92072 CF56SH 11995649 Ki = 112 nM T92072 C8FR7V 11995650 Ki = 96 nM T92072 C4YPA1 11995651 Ki = 16 nM T92072 CNX94G 12063014 Ki > 10000 nM T92072 CPF9I3 12066874 Ki = 79.43 nM T92072 CM8B4R 12293993 Ki = 34.8 nM T92072 CQ6TX7 12455201 Ki > 10000 nM T92072 CC8Q7D 12766586 Ki = 4620 nM T92072 CTE6H4 13155597 Ki = 3100 nM T92072 CWOQ92 13360944 Ki = 14800 nM T92072 CB4M0C 13506474 Ki = 9.2 nM T92072 C24VJF 13608091 Ki = 14 nM T92072 C97BVY 13830108 Ki = 0.67 nM T92072 CU25GH 14000479 Ki = 69 nM T92072 CVS4J0 14426726 Ki = 0.59 nM T92072 CM2XP1 14476141 EC50 = 8000 nM T92072 COU82X 14686957 Ki = 199.53 nM T92072 CCB92W 14686958 Ki = 3400 nM T92072 CP1QI6 14686969 Ki = 316.23 nM T92072 CR98ZM 14788199 Ki > 3000 nM T92072 CC96OF 14788202 Ki = 130 nM T92072 CI9JQ2 14788203 Ki = 90 nM T92072 C6KL1N 14788206 Ki = 41 nM T92072 C4BW2R 14788208 Ki = 20 nM T92072 C83SZT 14788210 Ki = 8 nM T92072 CM3I7A 14788211 Ki = 17 nM T92072 C28PEO 14788213 Ki = 85 nM T92072 CT2ON1 14788223 Ki = 8 nM T92072 CNC76O 14788224 Ki = 2.6 nM T92072 CS8YF3 14788225 Ki = 14 nM T92072 C0AI3P 14788226 Ki = 82 nM T92072 CN14KT 14788227 Ki > 10000 nM T92072 CAB8P0 14788228 Ki = 100 nM T92072 CG74UN 14788231 Ki = 76 nM T92072 CR4H7P 14788232 Ki = 53 nM T92072 CT6K9F 14788235 Ki = 660 nM T92072 CU6H7J 14788237 Ki = 11 nM T92072 CQS35H 14842888 Ki = 2060 nM T92072 C76FZJ 14873275 Ki > 10000 nM T92072 CQ7MK8 15388822 Ki = 3360 nM T92072 CSQ0R5 15388827 Ki = 3230 nM T92072 CEN2O9 15388828 Ki = 16300 nM T92072 CPD7A4 15588319 Ki > 10000 nM T92072 C65SCN 15599151 Ki = 0.76 nM T92072 CG0I8D 15667089 Ki = 2.2 nM T92072 C8OZ5G 15667105 Ki = 0.7 nM T92072 CE13QR 15729970 Ki = 138 nM T92072 CV8DE2 15729973 Ki = 1940 nM T92072 CFD31U 15729977 Ki = 4310 nM T92072 C31TPS 15950360 Ki = 2990 nM T92072 C3GP9F 15987727 Ki > 10000 nM T92072 C7H5ZS 15987740 Ki > 10000 nM T92072 CT9I7F 16036826 Ki = 1298 nM T92072 C2L4NO 16037920 IC50 = 183 nM T92072 C05KOS 16050635 Ki > 7500 nM T92072 CI32XZ 16064248 Ki = 236 nM T92072 C6UEW5 16064250 Ki = 8598 nM T92072 C6M3VK 16064568 Ki = 4640 nM T92072 C04WQF 16064570 Ki = 5138 nM T92072 CH72WU 16064711 Ki = 1800 nM T92072 C2Q9UM 16070216 Ki = 1040 nM T92072 C8Z2WO 16070220 Ki = 2254 nM T92072 C80TJF 16070335 Ki = 312 nM T92072 CWFS63 16071777 Ki = 11 nM T92072 C9K2PE 16071901 Ki = 25 nM T92072 CN7F9X 16072019 Ki = 454 nM T92072 CGX62B 16072020 Ki = 42 nM T92072 CL4ON2 16072021 Ki = 55 nM T92072 CU42YH 16072022 Ki = 17 nM T92072 CXS8C0 16072023 Ki = 18 nM T92072 CSO1T2 16072024 Ki = 98 nM T92072 C8W5EP 16087946 Ki = 110 nM T92072 CK29IS 16094546 Ki = 1000 nM T92072 C8B5YT 16094547 Ki = 848 nM T92072 CM94FD 16094548 Ki = 3800 nM T92072 C7FSA9 16094549 Ki = 1970 nM T92072 C9W2FV 16094550 Ki = 589 nM T92072 C32PKU 16094551 Ki = 1430 nM T92072 CF23NY 16094554 Ki = 770 nM T92072 CTB39W 16094555 Ki = 956 nM T92072 C8ZT6A 16094558 Ki = 750 nM T92072 C2VJ1H 16094559 Ki = 510 nM T92072 CA9QY7 16094561 Ki = 830 nM T92072 C18FPZ 16094562 Ki = 2920 nM T92072 C6BI2H 16094563 Ki = 1270 nM T92072 CBU5P4 16094566 Ki = 335 nM T92072 C3IX9U 16094567 Ki = 957 nM T92072 C9MO8F 16094568 Ki = 590 nM T92072 C7PJ9U 16094569 Ki = 1640 nM T92072 C8X6FC 16094570 Ki = 1250 nM T92072 C1E6YK 16094574 Ki = 429 nM T92072 C7DV1Q 16094575 Ki = 60 nM T92072 C6JML5 16100255 Ki = 590 nM T92072 C1T7DI 16103162 Ki > 5000 nM T92072 C87PRE 16103163 Ki > 5000 nM T92072 C34YIZ 16103164 Ki > 5000 nM T92072 C6U0TL 16103165 Ki = 1100 nM T92072 CT9O5K 16103166 Ki > 5000 nM T92072 CA2W9G 16103167 Ki = 3500 nM T92072 CG74XQ 16103168 Ki = 2600 nM T92072 CL87PX 16103169 Ki = 62 nM T92072 C01PWF 16103170 Ki > 5000 nM T92072 CO3HF4 16103171 Ki > 5000 nM T92072 CIAE42 16103176 Ki = 1050 nM T92072 C0Z4KU 16103177 Ki = 780 nM T92072 C3Y8IU 16103178 Ki = 700 nM T92072 CA1EH0 16103179 Ki > 5000 nM T92072 CJ8O9B 16103184 Ki = 933 nM T92072 CY3R6K 16103185 Ki = 737 nM T92072 C9F7SM 16103186 Ki = 1600 nM T92072 C7HM0K 16103187 Ki = 610 nM T92072 C9Q2MO 16109360 EC50 = 12.02 nM T92072 CR4GH8 16109369 EC50 = 0.7079 nM T92072 CGP93C 16115479 Ki = 901 nM T92072 CX4O9C 16115613 Ki = 53 nM T92072 CCZ67Y 16115614 Ki = 3990 nM T92072 C4TDQ5 16115615 Ki = 12000 nM T92072 C4EW6I 16115616 Ki = 3000 nM T92072 C4FI6K 16115617 Ki = 1880 nM T92072 CYKC87 16115749 Ki = 1420 nM T92072 C4A8SU 16115750 Ki = 1880 nM T92072 C8VXL9 16115751 Ki = 58 nM T92072 CRH54T 16115902 Ki = 153 nM T92072 C53DBK 16115903 Ki = 9140 nM T92072 CT5UQ7 16115904 Ki = 48100 nM T92072 CRZ0V4 16115905 Ki = 53800 nM T92072 CK87MV 16115906 Ki = 175 nM T92072 C3G6FA 16115907 Ki = 4090 nM T92072 CC53PW 16116048 Ki = 1230 nM T92072 C0S1VK 16122818 Ki = 410 nM T92072 CA49CN 16122819 Ki = 340 nM T92072 CHT26E 16202442 IC50 = 0.6761 nM T92072 CO8WS3 16203544 Ki = 579 nM T92072 CH91QO 16203667 Ki = 73.6 nM T92072 CTL0F3 16203668 Ki = 640 nM T92072 C4OS0D 16203669 Ki = 190 nM T92072 C0KL4A 16220189 Ki = 2490 nM T92072 CZT4J2 16433205 Ki > 100000 nM T92072 C4QU0M 16654984 Ki = 40 nM T92072 CFE82W 16656768 Ki = 6220 nM T92072 C7WF2V 16720104 Ki > 10000 nM T92072 CT7UO9 16720105 Ki > 10000 nM T92072 C9JSW0 16720106 Ki > 10000 nM T92072 C4T9HB 16735540 Ki = 55.4 nM T92072 CDV52Y 16739249 Ki = 379 nM T92072 CLU01J 16755701 Ki > 25000 nM T92072 C6PLG1 17035744 Ki = 11.6 nM T92072 CZX1Y3 17035750 Ki = 2.5 nM T92072 CBR05N 17198004 Ki = 20 nM T92072 CWD1N7 17429448 Ki = 1300 nM T92072 CXRL32 17863158 IC50 > 10000 nM T92072 CL9AX4 17863209 IC50 > 10000 nM T92072 CELB65 17863210 IC50 = 2600 nM T92072 CF87SP 18440405 Ki = 373 nM T92072 CX6J0D 18440417 Ki = 80 nM T92072 CRJ31X 18440425 Ki = 330 nM T92072 CKE94U 18440431 Ki = 2330 nM T92072 CZO7K8 18440528 Ki = 583 nM T92072 CH29ON 18440555 Ki = 3640 nM T92072 CQZ3E9 19003740 Ki = 42 nM T92072 CTS2L7 19003749 Ki = 22 nM T92072 C0VD9T 19574102 Ki = 3162.28 nM T92072 CL8U0R 20109827 EC50 = 12000 nM T92072 CBXA48 20592013 Ki = 1.87 nM T92072 C86NHU 20696356 EC50 = 28 nM T92072 CBC2U1 20770622 Ki = 1116 nM T92072 C5KR4S 20847387 Ki > 100000 nM T92072 C1N7ZG 20974732 Ki = 3200 nM T92072 CW50HY 20974734 Ki = 800 nM T92072 CM7C5Y 21180383 Ki = 7600 nM T92072 CPV9N1 21591949 Ki = 26 nM T92072 CB2V8H 21603068 Ki = 29700 nM T92072 C25WAJ 21874520 Ki = 1133 nM T92072 CTK29C 21874538 Ki = 291 nM T92072 C96PRF 21874571 Ki = 190 nM T92072 C07MZN 21874581 Ki = 319 nM T92072 C5QJC8 21874602 Ki = 733 nM T92072 CXG16I 21874603 Ki = 110 nM T92072 CV2C4F 21874613 Ki = 50 nM T92072 CB7S8A 21874626 Ki = 700 nM T92072 CKG68C 21874634 Ki = 1166 nM T92072 CTX5P2 21874639 Ki = 2965 nM T92072 C1CKS9 21874641 Ki = 249 nM T92072 CU80AG 21874647 Ki = 19 nM T92072 C38CXY 21874661 Ki = 120 nM T92072 C4S5PJ 21874662 Ki = 190 nM T92072 C14FGO 21874668 Ki = 77 nM T92072 C3WLM0 21874675 Ki = 27 nM T92072 COLC85 21874676 Ki = 118 nM T92072 C2PZN3 21874681 Ki = 40 nM T92072 CP84GK 21874685 Ki = 83 nM T92072 CSV0W4 21874686 Ki = 190 nM T92072 CW47EF 21874687 Ki = 931 nM T92072 C3EK0T 21874692 Ki = 769 nM T92072 C3KH4A 21874697 Ki = 42 nM T92072 CDV73C 21874721 Ki = 98 nM T92072 C7GWD4 21874722 Ki = 4909 nM T92072 C4L8UK 21874755 Ki = 4143 nM T92072 CLY0E3 21874756 Ki = 26 nM T92072 CWQ47T 21874764 Ki = 2531 nM T92072 C74HIZ 21874771 Ki = 230 nM T92072 C7NT1D 21874782 Ki = 117 nM T92072 CG9Y7N 21874786 Ki = 183 nM T92072 CK4HL6 21916357 Ki = 1480 nM T92072 CZRX51 21916371 Ki = 617 nM T92072 CS19AF 21916389 Ki = 185 nM T92072 CBY0E6 21916394 Ki = 218 nM T92072 CI1CO9 21916398 Ki = 352 nM T92072 CZ59CO 21916406 Ki = 167 nM T92072 C2XR0J 21916408 Ki = 347 nM T92072 C03FGL 21916419 Ki = 154 nM T92072 CB56UX 21958512 Ki = 305 nM T92072 CBA86P 21958522 Ki > 10000 nM T92072 C4I2HN 21958524 Ki = 3290 nM T92072 CKQ1C3 21958525 Ki > 6000 nM T92072 CBQF27 21958526 Ki = 6.4 nM T92072 CZ92NC 21958536 Ki = 76 nM T92072 CFX4B6 21958541 Ki = 5180 nM T92072 C2CFG0 21958557 Ki = 582 nM T92072 CZN1L8 21958583 Ki = 290 nM T92072 CW5NK7 21958593 Ki = 1800 nM T92072 C36FJO 21958619 Ki = 274 nM T92072 CJ7IB6 21958676 Ki = 643 nM T92072 CTSU04 21958681 Ki = 5600 nM T92072 CW5DG9 21958701 Ki = 102 nM T92072 C7RE2I 21958724 Ki = 416 nM T92072 CJO62E 21958725 Ki = 5100 nM T92072 C6F8TR 21958745 Ki > 6000 nM T92072 CMF03Z 21958758 Ki = 2600 nM T92072 C58MPT 21958761 Ki > 6000 nM T92072 C5L8YT 21958762 Ki = 178 nM T92072 C4K7OP 21958764 Ki = 275 nM T92072 CCTJ56 21958775 Ki = 210 nM T92072 CU7EZ3 21958783 Ki > 6000 nM T92072 CUNF42 21958814 Ki = 930 nM T92072 C5HFL6 22002319 Ki = 428 nM T92072 CFH75K 22002352 Ki = 958 nM T92072 C02SLQ 22002364 Ki = 315 nM T92072 CPS61Y 22002375 Ki = 135 nM T92072 C3CV9X 22002449 Ki = 185 nM T92072 CW24GQ 22015484 Ki = 1642 nM T92072 CEWY38 22015485 Ki = 47 nM T92072 CNJ90S 22015489 Ki = 497 nM T92072 CDUS06 22015491 Ki = 6321 nM T92072 C8M3PX 22015492 Ki = 4900 nM T92072 CDN7B6 22015493 Ki = 193 nM T92072 C6P2DA 22015494 Ki = 462 nM T92072 CD0KT8 22015499 Ki = 123 nM T92072 CJ0Z6F 22015500 Ki = 647 nM T92072 CN7O2U 22015504 Ki = 13 nM T92072 C05CGK 22015508 Ki = 320 nM T92072 CQ07MJ 22015509 Ki = 504 nM T92072 CG8Z5Y 22015516 Ki = 721 nM T92072 CV6F4T 22015525 Ki = 175 nM T92072 C48YPI 22015526 Ki = 1610 nM T92072 CQL6X2 22015529 Ki = 7255 nM T92072 CS8IX9 22015530 Ki = 779 nM T92072 C7RV4D 22015532 Ki = 206 nM T92072 CVH03D 22015533 Ki = 709 nM T92072 CYN5L0 22015535 Ki = 1605 nM T92072 CU41EO 22015539 Ki = 6219 nM T92072 CAU0Z3 22015549 Ki = 763 nM T92072 CPK81R 22015550 Ki = 468 nM T92072 CKME84 22055296 Ki = 100 nM T92072 C43TSO 22055299 Ki = 41 nM T92072 CE6U0L 22220610 Ki = 4.9 nM T92072 C67RYE 22252243 Ki = 8775 nM T92072 C7CW3I 22266730 Ki > 6000 nM T92072 CZF4S2 22266732 Ki > 6000 nM T92072 CTO91Z 22266738 Ki = 540 nM T92072 C75PVI 22266740 Ki > 6000 nM T92072 CC2N6M 22266741 Ki > 6000 nM T92072 CZL43T 22266742 Ki > 6000 nM T92072 C0XT6H 22266744 Ki = 348 nM T92072 CV6E4A 22266746 Ki = 260 nM T92072 CU16OK 22266751 Ki > 6000 nM T92072 C2QUH0 22266756 Ki > 6000 nM T92072 CLF81K 22266759 Ki > 6000 nM T92072 CIOB39 22266761 Ki = 3500 nM T92072 CC12SJ 22266763 Ki > 6000 nM T92072 C4ZJ1F 22266765 Ki = 1000 nM T92072 C3WK8Z 22266766 Ki > 6000 nM T92072 CAGC71 22266769 Ki = 2190 nM T92072 CV53YM 22266771 Ki > 6000 nM T92072 CSC37U 22266775 Ki = 1500 nM T92072 CCQ0I1 22266776 Ki = 1400 nM T92072 CDWI49 22266778 Ki = 427 nM T92072 CC94DE 22266784 Ki > 6000 nM T92072 C7G0LF 22282339 Ki > 666 nM T92072 CPDA63 22283414 Ki = 1600 nM T92072 CMF83X 22428505 Ki = 3200 nM T92072 CYP2Z4 22674365 Ki = 400 nM T92072 CL95BF 22674372 Ki = 487 nM T92072 CIHV23 22674379 Ki = 1364 nM T92072 CIK25F 22674386 Ki = 710 nM T92072 CJVG74 22674390 Ki = 14 nM T92072 CJ1H3A 22674393 Ki = 4216 nM T92072 CXV1G4 22674398 Ki = 295 nM T92072 CV3IJ9 22674410 Ki = 107 nM T92072 C0ITC9 22674411 Ki = 32 nM T92072 CQ16FW 22674422 Ki > 100000 nM T92072 C54ZKH 22674428 Ki = 33 nM T92072 CZS72H 22674456 Ki = 1458 nM T92072 C4PK7T 22674477 Ki = 1733 nM T92072 CE7FI3 22674484 Ki = 5462 nM T92072 C1T3OA 22674492 Ki = 3474 nM T92072 CJ52EV 23371936 Ki > 100000 nM T92072 CFT0A1 23371944 Ki > 100000 nM T92072 C6OCL1 23546899 Ki = 1953 nM T92072 C8IU6O 23653582 EC50 > 3000 nM T92072 C65SJK 23656931 Ki = 65.2 nM T92072 CGRT64 23656932 Ki = 46 nM T92072 C8N0LF 23656933 Ki = 106.7 nM T92072 CYU94Z 23656934 Ki = 204.5 nM T92072 C8SC3A 23656935 Ki = 389.2 nM T92072 CO98NZ 23656936 Ki = 80.9 nM T92072 CV28WL 23656937 Ki = 916 nM T92072 CAG3Y8 23657103 Ki = 116.5 nM T92072 CKRG98 23657104 Ki = 462.2 nM T92072 C6YS2Z 23657105 Ki = 43.9 nM T92072 CZ6H4G 23657106 Ki = 104.2 nM T92072 C6F4UV 23657107 Ki = 89.5 nM T92072 C26AWG 23657108 Ki = 80.2 nM T92072 C0R9DW 23657109 Ki = 19 nM T92072 COD51S 23657262 Ki = 99 nM T92072 CSZB58 23657263 Ki > 10000 nM T92072 C68QBD 23657264 Ki = 256 nM T92072 C1SWM6 23657265 Ki = 2700 nM T92072 CG4I1H 23657266 Ki > 10000 nM T92072 CMSG38 23657267 Ki = 91.1 nM T92072 C6GDP9 23657408 Ki = 764 nM T92072 CVBI12 23657409 Ki > 10000 nM T92072 CFE2N1 23757284 Ki = 2.1 nM T92072 CVO53U 23900137 Ki = 1.9 nM T92072 C63GJC 24464119 Ki = 3090.3 nM T92072 CG8BZ4 24739307 Ki = 68 nM T92072 C1SGW5 24739308 Ki = 270 nM T92072 CFVO28 24739309 Ki = 120 nM T92072 CU12PX 24739310 Ki = 100 nM T92072 CK96FD 24739478 Ki = 150 nM T92072 CJ23NC 24739479 Ki = 1400 nM T92072 CUW7F4 24739481 Ki = 200 nM T92072 CG95TO 24739646 Ki = 68 nM T92072 C5JK9I 24739647 Ki = 600 nM T92072 CO46JZ 24739648 Ki = 78 nM T92072 CQ5H6Y 24739649 Ki = 540 nM T92072 COB5Q7 24739812 Ki = 120 nM T92072 C1Y7AV 24739813 Ki = 480 nM T92072 CRN05P 24739814 Ki = 140 nM T92072 CRT41U 24768400 Ki = 218 nM T92072 C3EVZ7 24768401 Ki = 1700 nM T92072 CIU04J 24768402 Ki = 850 nM T92072 C8I3OV 24768403 Ki = 390 nM T92072 C7RGV4 24768404 Ki = 850 nM T92072 C2PRD9 24768405 Ki = 389 nM T92072 CS7M9E 24768406 Ki = 4200 nM T92072 C3NO0Z 24768407 Ki = 1700 nM T92072 CJD61X 24768408 Ki > 10000 nM T92072 C5X9OD 24768409 Ki > 10000 nM T92072 CF6BC7 24768410 Ki = 850 nM T92072 CAG7S1 24768411 Ki = 930 nM T92072 CAG8R2 24768412 Ki = 4400 nM T92072 CSL71N 24768413 Ki = 1998 nM T92072 CJ2V9Z 24768414 Ki = 1880 nM T92072 CZ4J5K 24768415 Ki = 2100 nM T92072 CQ63KX 24768416 Ki = 890 nM T92072 C8OGP3 24768417 Ki = 71 nM T92072 C4ZRC9 24768418 Ki = 380 nM T92072 C1A0NS 24768419 Ki = 540 nM T92072 C35QUL 24768420 Ki = 500 nM T92072 C6XR5O 24768421 Ki = 630 nM T92072 CAG3S6 24768422 Ki = 1210 nM T92072 CI6B4H 24768423 Ki = 1020 nM T92072 CXEC07 24768424 Ki = 347 nM T92072 CS0C6Q 24768425 Ki = 940 nM T92072 C3E6MK 24768426 Ki = 262 nM T92072 C46NSY 24768427 Ki = 2300 nM T92072 CF8C0L 24768428 Ki = 270 nM T92072 CBMC42 24768429 Ki = 370 nM T92072 CR5H8A 24768430 Ki = 2600 nM T92072 CA3UK5 24768431 Ki = 550 nM T92072 CG8QK3 24768432 Ki = 220 nM T92072 CMT5N1 24768433 Ki = 210 nM T92072 C6HW8J 24768434 Ki = 630 nM T92072 CS85OX 24768440 Ki = 486 nM T92072 C2U5TQ 24768441 Ki = 5474 nM T92072 CGVO15 24768442 Ki = 1462 nM T92072 CSJW71 24768444 Ki = 2445 nM T92072 C53BPO 24768445 Ki = 1840 nM T92072 CYZI26 24768446 Ki = 582 nM T92072 C90QOD 24768449 Ki = 2443 nM T92072 C06UBG 24768450 Ki = 2080 nM T92072 C09WQS 24768452 Ki = 4480 nM T92072 C6ZDA2 24778159 Ki = 28 nM T92072 C6S1HG 24810000 Ki = 9 nM T92072 CK02ZF 24812771 Ki = 162 nM T92072 CGH0U3 24827290 Ki = 420 nM T92072 C5UO3Z 24827415 Ki = 350 nM T92072 C32BCU 24827417 Ki = 370 nM T92072 CKC0W3 24827442 Ki = 631 nM T92072 C0WA2D 24827443 Ki = 410 nM T92072 CQW7H1 24827444 Ki = 522 nM T92072 CIR6E9 24827552 Ki = 1520 nM T92072 C15VIG 24827553 Ki = 2500 nM T92072 C06PBV 24827554 Ki = 3590 nM T92072 C34RNS 24827555 Ki = 1280 nM T92072 CGUY42 24827556 Ki = 1120 nM T92072 C2W7YS 24828056 Ki = 376 nM T92072 CWPS95 24828457 Ki = 1200 nM T92072 CU0Q2I 24878975 Ki > 10000 nM T92072 C05BYL 24882472 Ki = 356 nM T92072 C8DTC3 24894065 Ki = 406 nM T92072 C0PHN9 24939231 Ki = 1.2 nM T92072 C0WF2D 24950372 Ki = 48 nM T92072 C47TZM 24950529 Ki = 68 nM T92072 CY5W4G 24950531 Ki = 34 nM T92072 C31DGI 24950532 Ki = 250 nM T92072 CU24RD 24950533 Ki = 11 nM T92072 CE75OM 24950689 Ki = 270 nM T92072 C45DXE 24950690 Ki = 64 nM T92072 C6PT5O 24950691 Ki = 34 nM T92072 CS1ZM6 24950846 Ki = 100 nM T92072 CZK1X7 24989636 Ki = 913 nM T92072 CWPX23 24989637 Ki = 4954 nM T92072 C03WIO 24989638 Ki = 2473 nM T92072 C0YGQ2 24998410 Ki = 11700 nM T92072 C2EK5G 25002987 Ki = 1430 nM T92072 COSA97 25003338 Ki = 860 nM T92072 C7DF0O 25003339 Ki = 790 nM T92072 C1ZXW0 25003340 Ki = 530 nM T92072 CHEX21 25003341 Ki = 1150 nM T92072 CL5NI4 25008276 IC50 >= 10000 nM T92072 CW5YA6 25066016 Ki = 259 nM T92072 CX43GT 25069599 Ki = 4600 nM T92072 CP3Y5K 25069603 Ki = 440 nM T92072 CM1WB9 25069914 Ki = 130 nM T92072 CK92QL 25070230 Ki = 10 nM T92072 C04QRE 25074004 Ki = 55 nM T92072 C07GFA 25074313 Ki = 220 nM T92072 CLWN54 25074316 Ki = 77.2 nM T92072 C2X4WJ 25099116 Ki = 50.12 nM T92072 CI9MP1 25099163 Ki = 5.754 nM T92072 CX63TW 25129539 Ki = 1070 nM T92072 C04QUH 25130167 EC50 = 7100 nM T92072 C1R6DV 25130168 EC50 = 7100 nM T92072 CFG50N 25130169 EC50 = 13000 nM T92072 C5U0BT 25130170 EC50 = 2500 nM T92072 C6Q9EF 25130523 EC50 = 8400 nM T92072 CD78XN 25130524 EC50 = 4900 nM T92072 C3YH5W 25138072 Ki = 290 nM T92072 CMP7V1 25138073 Ki = 2100 nM T92072 CLW7O5 25138074 Ki = 820 nM T92072 C7L6SP 25138075 Ki = 65 nM T92072 C1PF5O 25138076 Ki = 110 nM T92072 CC4HW2 25138077 Ki = 22 nM T92072 C9J1MQ 25138078 Ki = 190 nM T92072 C9LMW0 25138079 Ki = 195 nM T92072 C2QLK4 25138080 Ki = 110 nM T92072 CS89DE 25138081 Ki = 940 nM T92072 C5AJ0V 25138082 Ki = 70 nM T92072 CAL52B 25138083 Ki = 780 nM T92072 CZ41XS 25138084 Ki = 620 nM T92072 CA7JE4 25138085 Ki = 580 nM T92072 C9GZ6D 25138086 Ki = 81 nM T92072 C5A1FW 25138087 Ki = 7.2 nM T92072 CZ49VH 25138088 Ki = 31 nM T92072 CA01RE 25138089 Ki = 280 nM T92072 CC5O4P 25138090 Ki = 120 nM T92072 CQ30KW 25138091 Ki = 34 nM T92072 CCM9X1 25138092 Ki = 470 nM T92072 C7JE1V 25147618 Ki > 1000 nM T92072 C5FHU3 25147619 Ki > 1000 nM T92072 CN2FL7 25188209 Ki = 599 nM T92072 C1O2VJ 25207955 Ki = 323 nM T92072 CD2BJ5 25207956 Ki = 1037 nM T92072 C5J0UG 25207957 Ki = 2934 nM T92072 C5ZHT9 25207959 Ki = 320 nM T92072 C1YWI8 25207960 Ki = 4468 nM T92072 CJ8LD2 25207961 Ki = 4186 nM T92072 CHT85D 25208107 Ki = 64 nM T92072 CL7UJ3 25208108 Ki = 12100 nM T92072 CL5JR6 25208109 Ki = 352 nM T92072 C8RW4K 25208254 Ki = 620 nM T92072 CXK1G5 25208255 Ki = 215 nM T92072 CR6O3B 25208256 Ki = 325 nM T92072 CA3LY1 25208257 Ki = 150 nM T92072 C6TI7Y 25208258 Ki = 69 nM T92072 C2WT8G 25208259 Ki = 64 nM T92072 CN9XE6 25208260 Ki = 960 nM T92072 CHG1N9 25209990 Ki = 125 nM T92072 C0IBC5 25209991 Ki = 10.5 nM T92072 CFT98K 25210116 Ki = 203 nM T92072 CYK7O5 25210117 Ki = 354 nM T92072 CEYP97 25210118 Ki = 92 nM T92072 CZ3E6O 25210119 Ki = 1283 nM T92072 C7MI5W 25210254 Ki = 4466 nM T92072 C74JQH 25210255 Ki = 3364.3 nM T92072 COF2H0 25210256 Ki = 8124 nM T92072 C7T6PR 25210257 Ki > 10000 nM T92072 CI01GB 25211166 Ki > 10000 nM T92072 CU6OR2 25211167 Ki = 1460 nM T92072 C6S0OK 25242240 Ki = 2.4 nM T92072 CJ4K1Z 25242440 Ki = 58.4 nM T92072 CI1GW6 25268841 Ki = 48.2 nM T92072 C5HG7N 25553043 Ki = 2818.38 nM T92072 CEG8X7 28622387 Ki = 35 nM T92072 CS0V9B 32178888 Ki = 3700 nM T92072 C8DT0B 32459044 Ki = 1500 nM T92072 C4MB8S 32460014 Ki = 3300 nM T92072 C3FH2I 32460336 Ki = 1100 nM T92072 C6LI7R 32460717 Ki = 500 nM T92072 CU51PG 32461094 Ki = 2300 nM T92072 C4OUE0 32461100 Ki = 1600 nM T92072 C8TE4D 32461405 Ki = 5200 nM T92072 CKS89N 32461556 Ki = 3900 nM T92072 C40SYI 32866639 Ki = 3715.35 nM T92072 CVD0Q4 32867716 Ki = 2951.21 nM T92072 C4WD8U 39079816 EC50 = 4400 nM T92072 CWUA82 42625614 Ki = 28.4 nM T92072 C6W4XM 42625615 Ki = 12.8 nM T92072 CX8DV9 42625691 Ki = 1680 nM T92072 C5I8NE 42625766 Ki = 258 nM T92072 CIG29P 42625767 Ki = 2150 nM T92072 C4NS7C 42625924 Ki = 114 nM T92072 C4RHY0 42630191 IC50 = 150 nM T92072 CDSI21 42631399 Ki > 100000 nM T92072 C5YV2R 42631400 Ki = 11200 nM T92072 CP31OD 42631506 Ki = 43000 nM T92072 CKEC01 42631507 Ki > 100000 nM T92072 CBJ07K 42631609 Ki = 800 nM T92072 C1QS2X 42631610 Ki = 2100 nM T92072 CVX80U 42631613 Ki > 100000 nM T92072 C6SVP2 42631614 Ki > 100000 nM T92072 C0O1HM 42631715 Ki > 100000 nM T92072 C3M5GK 42631719 Ki = 13500 nM T92072 C0EYB8 42631813 Ki > 100000 nM T92072 C0UH7I 42631818 Ki = 14000 nM T92072 CT57MJ 42631819 Ki = 2100 nM T92072 CS0O4J 42631924 Ki = 1600 nM T92072 CTBW80 42636897 Ki = 0.51 nM T92072 CK43JX 44157013 Ki = 1967 nM T92072 C1J6SG 44185870 Ki > 1000 nM T92072 CX24EI 44185874 Ki > 10000 nM T92072 CWX1B7 44185933 Ki > 10000 nM T92072 C8I9LD 44185936 Ki = 1170 nM T92072 CQRH91 44186579 Ki = 1840 nM T92072 C9RG0P 44186580 Ki > 10000 nM T92072 CCNH98 44186622 Ki = 1090 nM T92072 CY2D4F 44186623 Ki = 1820 nM T92072 CAY95F 44186625 Ki = 2070 nM T92072 C42DUI 44186626 Ki = 2300 nM T92072 CYE0X8 44186667 Ki = 5630 nM T92072 CM7B3X 44186668 Ki = 2300 nM T92072 C69VCO 44186669 Ki = 2610 nM T92072 C5X9NC 44186716 Ki = 3800 nM T92072 C6JG3Q 44186717 Ki > 10000 nM T92072 CE21OP 44186718 Ki > 10000 nM T92072 C9W0OQ 44186719 Ki = 443 nM T92072 C59XNK 44203236 Ki = 3760 nM T92072 CIL82A 44203643 Ki = 36.9 nM T92072 CE6C9F 44203644 Ki = 85.7 nM T92072 C6I4TU 44217536 Ki = 1405 nM T92072 CG5BH8 44218327 Ki = 1398 nM T92072 C0SBK7 44232535 Ki = 14900 nM T92072 CK1H5B 44241696 Ki = 346 nM T92072 CD2I6F 44276002 EC50 = 2890 nM T92072 CP5M2R 44276273 EC50 = 2280 nM T92072 C7T0ZY 44281663 Ki = 1725 nM T92072 CX3YV9 44281684 Ki > 1000 nM T92072 CJ3QM8 44281700 Ki = 1361 nM T92072 CN72HK 44281738 Ki = 1175 nM T92072 C7HV4D 44284007 Ki = 5450 nM T92072 CL8XS1 44284052 Ki = 733 nM T92072 C28QCM 44284065 Ki = 1620 nM T92072 C8YHM6 44284095 Ki = 432 nM T92072 CUR2Q6 44284189 Ki = 342 nM T92072 CE5V1M 44284209 Ki = 31.8 nM T92072 CBQ90F 44284222 Ki = 252 nM T92072 C34FVI 44284223 Ki = 207 nM T92072 CT0EV8 44284345 Ki = 70.7 nM T92072 C4PT0D 44297686 Ki = 971 nM T92072 CRAW93 44299582 Ki = 50 nM T92072 C7O5MJ 44309799 EC50 > 10000 nM T92072 CCQ4Y0 44317558 Ki = 951 nM T92072 CW93LX 44317576 Ki = 132 nM T92072 CW1G8S 44317578 Ki = 144 nM T92072 C1RFW2 44317916 Ki = 771 nM T92072 CJS3C0 44317969 Ki = 896 nM T92072 CI7RG8 44317970 IC50 = 5647 nM T92072 CZQ51K 44323390 Ki = 8 nM T92072 CY1SP3 44324421 IC50 = 9 nM T92072 CV9NA5 44324599 IC50 = 2500 nM T92072 C8T0GE 44327984 Ki = 100 nM T92072 C2WU1X 44333135 Ki > 10000 nM T92072 C6ALX7 44333187 Ki = 1995.26 nM T92072 CVGR26 44333267 Ki > 10000 nM T92072 C1SVU5 44333456 Ki > 10000 nM T92072 CGTS60 44333467 Ki > 10000 nM T92072 CDQ9I3 44337955 IC50 = 3.9 nM T92072 C2U4CB 44343895 EC50 = 630.96 nM T92072 C8V6QA 44344926 Ki = 4600 nM T92072 CF28PI 44366534 Ki = 226 nM T92072 COK3D2 44366548 Ki = 321 nM T92072 CWM42Q 44366549 Ki = 72 nM T92072 CFS1R2 44366557 Ki = 1826 nM T92072 C97QUH 44366570 Ki = 253 nM T92072 CU84PA 44366586 Ki = 584 nM T92072 CJ5G0X 44366646 Ki = 524 nM T92072 CO3UB5 44366647 Ki = 238 nM T92072 C4G3NR 44366738 Ki = 12 nM T92072 C4ARH3 44366739 Ki = 1913 nM T92072 CRC4G6 44366748 Ki = 45 nM T92072 CP17RQ 44366753 Ki = 35 nM T92072 C52WVN 44366765 Ki = 71 nM T92072 CZ7IT8 44366857 Ki = 157 nM T92072 C2CJ4T 44366858 Ki = 306 nM T92072 CLO08W 44366860 Ki = 148 nM T92072 CZ4LC6 44366934 Ki = 140 nM T92072 CZK9I1 44366935 Ki = 96 nM T92072 CPSY05 44366944 Ki = 205 nM T92072 CLPK45 44366986 Ki = 167 nM T92072 CF43MH 44367050 Ki = 33 nM T92072 CIZ76P 44367051 Ki = 55 nM T92072 CIFK18 44367052 Ki = 235 nM T92072 CRDU48 44367064 Ki = 36 nM T92072 CV64BY 44367065 Ki = 209 nM T92072 C0LP4H 44367070 Ki = 50 nM T92072 C8U7JM 44367078 Ki = 78 nM T92072 C1NVX3 44367081 Ki = 1409 nM T92072 CF0Y5U 44367082 Ki = 157 nM T92072 CV32ZG 44374566 EC50 = 869 nM T92072 CE0GW9 44379809 Ki = 1900 nM T92072 CLU60V 44379847 Ki = 100 nM T92072 C80YID 44379848 Ki = 1800 nM T92072 CEQ85H 44379977 Ki = 2500 nM T92072 CX37RK 44380025 Ki = 7300 nM T92072 C4I3HP 44380110 Ki = 900 nM T92072 C53IPV 44380120 Ki = 6100 nM T92072 CY4DQ7 44390444 Ki > 6000 nM T92072 C3D6LX 44390522 Ki > 6000 nM T92072 CF6WX2 44390523 Ki = 113 nM T92072 C25RFG 44390527 Ki = 2010 nM T92072 CWR5M2 44390528 Ki = 1170 nM T92072 CBZ2P1 44390545 Ki = 8 nM T92072 CEB5I3 44390547 Ki > 6000 nM T92072 CE53OI 44390549 Ki > 6000 nM T92072 CG4KO6 44390551 Ki > 6000 nM T92072 CHZ5D1 44390559 Ki = 473 nM T92072 C6HBX7 44390571 Ki > 6000 nM T92072 C6XV9J 44390583 Ki > 6000 nM T92072 CLQ41H 44390587 Ki > 6000 nM T92072 CA4KL8 44390599 Ki > 6000 nM T92072 C0XIJ4 44390615 Ki > 6000 nM T92072 CD2F9O 44390651 Ki = 288 nM T92072 C8Q9XH 44390669 Ki > 6000 nM T92072 C83KXG 44396444 Ki > 5000 nM T92072 C7K1ST 44396450 Ki = 3800 nM T92072 C4AOY9 44396470 Ki = 4200 nM T92072 C32JTS 44396478 Ki = 1800 nM T92072 CHY08U 44396487 Ki = 4500 nM T92072 CS0D8B 44396500 Ki = 2000 nM T92072 C8B1XJ 44396515 Ki > 6000 nM T92072 CXZ7Q4 44396516 Ki = 770 nM T92072 CY7B3D 44396545 Ki > 4000 nM T92072 C7ERK1 44396546 Ki = 3000 nM T92072 C0N1FZ 44396599 Ki = 1300 nM T92072 CHT68B 44397718 Ki = 3170 nM T92072 C4TU8O 44397776 Ki = 34000 nM T92072 CJW4Q7 44398644 EC50 = 8800 nM T92072 CQ08PC 44398695 EC50 > 10000 nM T92072 C0WCS7 44398928 EC50 > 10000 nM T92072 C3EXH2 44398965 EC50 = 18200 nM T92072 C4QNR0 44401051 Ki = 0.8 nM T92072 CXCE96 44401487 Ki = 120 nM T92072 C5U2YX 44401545 Ki = 42 nM T92072 CT7W3U 44401604 Ki = 480 nM T92072 CQM65U 44402195 Ki = 3250 nM T92072 CXHS76 44402758 Ki = 2840 nM T92072 CV8BG5 44402784 Ki = 224 nM T92072 CFR09M 44403549 Ki > 10000 nM T92072 CDX4H0 44403550 Ki > 10000 nM T92072 C14IUF 44403555 Ki = 6240 nM T92072 CK2NB5 44403556 Ki = 630 nM T92072 C3QA1H 44403590 Ki > 10000 nM T92072 C8QT7Y 44403599 Ki > 10000 nM T92072 CB89RY 44403600 Ki > 10000 nM T92072 C6MWR3 44403601 Ki = 4160 nM T92072 CR06AD 44403609 Ki = 630 nM T92072 COKU07 44403611 Ki > 10000 nM T92072 C5CZ7U 44403618 Ki > 10000 nM T92072 C5WED3 44403621 Ki > 10000 nM T92072 C4C1WB 44403622 Ki = 5600 nM T92072 CMYR63 44403623 Ki > 10000 nM T92072 CU1BD7 44403629 Ki = 1650 nM T92072 C3EF0B 44403630 Ki = 4370 nM T92072 CV16HJ 44403635 Ki = 1580 nM T92072 CK73CA 44403636 Ki = 730 nM T92072 CG5HM3 44403643 Ki = 300 nM T92072 CA54QX 44403644 Ki = 717 nM T92072 CTE46U 44405094 Ki = 0.48 nM T92072 CB3X0L 44405124 Ki = 46 nM T92072 CN94AX 44406328 Ki = 2000 nM T92072 C3JPG9 44406334 Ki = 3300 nM T92072 C3S9CP 44406397 Ki = 4600 nM T92072 CAF1Y3 44406398 Ki = 3700 nM T92072 CT21RA 44406403 Ki = 3500 nM T92072 CA8FV4 44406545 Ki = 2500 nM T92072 CG8MQ9 44406555 Ki = 1900 nM T92072 CUPC05 44406556 Ki = 3000 nM T92072 C5ZW8S 44406562 Ki = 2200 nM T92072 CQ98MC 44406567 Ki = 1900 nM T92072 CN7V0Y 44406570 Ki = 3900 nM T92072 CI19OT 44406582 Ki = 1400 nM T92072 CZPM65 44406588 Ki = 810 nM T92072 C6O9TH 44406592 Ki = 530 nM T92072 CJA23V 44406607 Ki = 630 nM T92072 CV5AO7 44406611 Ki = 570 nM T92072 CE3CP9 44406617 Ki = 3500 nM T92072 CVQ2B8 44406625 Ki = 3000 nM T92072 CD9E7F 44406639 Ki = 3300 nM T92072 CK7GF1 44406642 Ki = 1300 nM T92072 CPEV01 44406643 Ki = 652 nM T92072 CK9ZB7 44407518 Ki > 10000 nM T92072 CES29R 44408316 Ki = 800 nM T92072 C0EB9D 44410399 Ki = 280 nM T92072 C6E4RA 44410402 Ki = 34.4 nM T92072 C5IVA3 44410403 Ki = 44.2 nM T92072 CI7W8R 44410406 Ki = 5.59 nM T92072 CWQX21 44410409 Ki = 4.27 nM T92072 CJ26LR 44410410 Ki = 716 nM T92072 CG30RK 44410412 Ki = 176 nM T92072 CK8I1V 44410544 Ki = 109 nM T92072 CO2LJ0 44410545 Ki = 19.9 nM T92072 CX9OZ0 44410549 Ki = 51.6 nM T92072 C7DER1 44410550 Ki = 3.47 nM T92072 C6E8OT 44410551 Ki = 4.24 nM T92072 CZ94PN 44410554 Ki = 11.3 nM T92072 COWL13 44410555 Ki = 15.5 nM T92072 CHU6Q0 44410556 Ki = 7.98 nM T92072 CVYF89 44410559 Ki = 131 nM T92072 C2YF8L 44410561 Ki = 6.11 nM T92072 CXD2R9 44410566 Ki = 1.24 nM T92072 C20FJQ 44410585 Ki = 65.3 nM T92072 CQ8E2B 44410597 Ki = 1.52 nM T92072 CYG5K3 44410655 Ki = 87 nM T92072 C41KLQ 44410684 Ki = 69.6 nM T92072 C8DE9A 44410690 Ki = 2.8 nM T92072 CSTP07 44410691 Ki = 3.12 nM T92072 CV37TH 44410697 Ki = 6.81 nM T92072 CV9C5B 44413096 IC50 = 140 nM T92072 CNDQ05 44413106 IC50 = 370 nM T92072 C7PAD9 44413113 IC50 = 350 nM T92072 C4QER5 44413125 IC50 = 126 nM T92072 C1PI5R 44413182 IC50 = 101 nM T92072 CMT4W9 44413192 IC50 = 12 nM T92072 C2ZH7P 44413202 IC50 = 102 nM T92072 COD4F9 44417680 Ki = 12 nM T92072 CM10LW 44420100 Ki = 840 nM T92072 CND70C 44420101 Ki = 218 nM T92072 CSR4Q2 44420921 Ki = 174 nM T92072 CWJ19B 44420922 Ki = 280 nM T92072 CO68UH 44420926 Ki = 7 nM T92072 CUE35G 44420928 Ki = 1560 nM T92072 C1V0HC 44420930 Ki = 331 nM T92072 C01VYU 44420931 Ki = 312 nM T92072 CX56TZ 44421598 Ki = 50.12 nM T92072 CE45HL 44421599 Ki = 5.012 nM T92072 CEH3F8 44421600 Ki = 100 nM T92072 C1NV4K 44421601 Ki = 50.12 nM T92072 C2C6DB 44421628 Ki = 251.19 nM T92072 C3C8LS 44423811 Ki = 8.5 nM T92072 CWCH32 44423812 Ki = 2.3 nM T92072 CDY6P7 44423813 Ki = 3.1 nM T92072 CYR14N 44423814 Ki = 3.5 nM T92072 C2F3DE 44423815 Ki = 5.2 nM T92072 CF26JD 44423816 Ki = 31.6 nM T92072 CE76XB 44423817 Ki = 4.7 nM T92072 C5J3PM 44423818 Ki = 7.7 nM T92072 CA2HW6 44423819 Ki = 15.3 nM T92072 CFM1I4 44423820 Ki = 8.4 nM T92072 CFTE30 44423821 Ki = 18.6 nM T92072 CQL6J8 44423822 Ki = 77.5 nM T92072 C4QFX3 44423823 Ki = 11.2 nM T92072 CWQK67 44423824 Ki = 20.4 nM T92072 CG5O9I 44423825 Ki = 28.3 nM T92072 CK1EQ6 44423826 Ki = 16.2 nM T92072 C4ZL9F 44423827 Ki = 30.5 nM T92072 CH96WQ 44423828 Ki = 50.4 nM T92072 CLJ9T4 44423837 Ki = 22.6 nM T92072 CT1YQ4 44423838 Ki = 30.8 nM T92072 C49JVO 44427579 Ki = 14 nM T92072 CID63L 44427580 Ki = 357 nM T92072 CWL9P8 44427581 Ki = 32 nM T92072 CG5C8V 44427582 Ki = 203 nM T92072 CVA8F6 44427583 Ki = 455 nM T92072 CGM8E6 44427584 Ki = 2875 nM T92072 C7L2KY 44427585 Ki = 57 nM T92072 C3Q1BN 44427586 Ki = 629 nM T92072 C91TWO 44427587 Ki = 250 nM T92072 CX1KI5 44427588 Ki = 60 nM T92072 C6BPF4 44427590 Ki = 201 nM T92072 C4FLS1 44427591 Ki = 559 nM T92072 C1GY3X 44427595 Ki = 6800 nM T92072 C7PT2S 44430151 Ki = 1300 nM T92072 CBW73G 44430154 Ki = 3 nM T92072 CDU4P8 44430156 Ki = 23 nM T92072 CA9L1D 44430158 Ki = 10 nM T92072 C9M0OF 44430160 Ki = 10 nM T92072 C0HBJ8 44430163 Ki = 24 nM T92072 CQF30M 44430165 Ki = 2 nM T92072 C2F3ZV 44430169 Ki = 43 nM T92072 C4IT7U 44430170 Ki = 27 nM T92072 C4S5DC 44430171 Ki = 6 nM T92072 CYS8I1 44430173 Ki = 8 nM T92072 CLW6M5 44430177 Ki = 1 nM T92072 CZ2CX5 44430187 Ki = 3 nM T92072 C42LMQ 44430188 Ki = 1 nM T92072 C0UDY1 44430192 Ki = 0.4 nM T92072 C87TZB 44430198 Ki = 74 nM T92072 CI97LW 44430203 Ki = 31 nM T92072 CPW14D 44430206 Ki = 36 nM T92072 CNX54A 44430209 Ki = 134 nM T92072 CC20AB 44430231 Ki = 39 nM T92072 C09MBQ 44430232 Ki = 20 nM T92072 CDH26R 44430235 Ki = 160 nM T92072 C8UN2W 44430236 Ki = 64 nM T92072 C07JTM 44430237 Ki = 1060 nM T92072 CX5RU6 44430239 Ki = 121 nM T92072 CL6C1D 44430241 Ki = 89 nM T92072 C41XMS 44435352 IC50 = 5.3 nM T92072 CLA42W 44435353 IC50 = 1.9 nM T92072 CATF75 44435354 IC50 = 380 nM T92072 CUFC32 44435355 IC50 = 85 nM T92072 C60SDL 44435356 IC50 = 3.2 nM T92072 CS7P6L 44435357 IC50 = 35 nM T92072 C08PCX 44435358 IC50 = 2.5 nM T92072 C18ANC 44435359 IC50 = 68 nM T92072 C3GB1N 44435360 IC50 = 254 nM T92072 CYP61J 44435361 IC50 = 9 nM T92072 C1TB8X 44436079 EC50 > 3000 nM T92072 CNX39I 44436082 EC50 > 3000 nM T92072 C21UTJ 44437214 Ki >= 25000 nM T92072 CAO98V 44437220 Ki > 25000 nM T92072 C67ZNA 44437460 Ki > 10000 nM T92072 CYB86Z 44442015 Ki = 290 nM T92072 C1UIO8 44442016 Ki = 1580 nM T92072 CUP5T0 44442018 Ki = 40 nM T92072 C4RDK6 44442019 Ki = 32 nM T92072 CPC63E 44442162 Ki = 100 nM T92072 C71XQS 44442163 Ki = 50 nM T92072 C42ZRD 44442166 Ki = 15 nM T92072 C9Z3CW 44442167 Ki = 7 nM T92072 C06RLU 44446477 Ki > 6000 nM T92072 CFPZ19 44447519 Ki = 1118 nM T92072 CJ7MS5 44447534 Ki = 4770 nM T92072 C3LOJ1 44447535 Ki = 837 nM T92072 C95AWU 44448014 Ki = 410 nM T92072 CL3WE0 44448018 Ki = 650 nM T92072 C3KQS2 44448019 Ki = 1100 nM T92072 CGYJ03 44448021 Ki = 2200 nM T92072 CU02SC 44448022 Ki = 1300 nM T92072 CYD75N 44448023 Ki = 4300 nM T92072 CTAH78 44448024 Ki = 1500 nM T92072 CMJ65Z 44448025 Ki = 2100 nM T92072 CHA97I 44448026 Ki = 9700 nM T92072 CX64PJ 44448028 Ki = 25000 nM T92072 CRU9L2 44448032 Ki = 180 nM T92072 C9I0XB 44448036 Ki = 87 nM T92072 C4NM9H 44448051 Ki = 73 nM T92072 CQ6BZ5 44448052 Ki = 270 nM T92072 CRO52K 44448053 Ki = 1200 nM T92072 C9FIN4 44448055 Ki = 95 nM T92072 CAOB06 44448056 Ki = 740 nM T92072 C64RXH 44448951 Ki = 271 nM T92072 C6SF2I 44448952 Ki = 181 nM T92072 C05ZJG 44448978 Ki = 265 nM T92072 CJ4DM9 44448979 Ki = 320 nM T92072 C74XLS 44448982 Ki = 454 nM T92072 CVEX70 44449007 Ki = 482 nM T92072 CJ8N1Z 44449034 Ki = 1040 nM T92072 CPL2F0 44449058 Ki = 160 nM T92072 CJLF50 44449113 Ki = 174 nM T92072 CP7Z2O 44449141 Ki = 3070 nM T92072 C2UWA8 44449279 Ki = 1993 nM T92072 CR4Z0Q 44449308 Ki = 1126 nM T92072 C8J0NG 44449493 Ki = 2726 nM T92072 CV63AZ 44449494 Ki = 748 nM T92072 CKL58O 44449520 Ki = 547 nM T92072 C60TLI 44449522 Ki = 835 nM T92072 CME34Q 44449532 Ki = 14 nM T92072 CL4HT0 44449533 Ki = 250 nM T92072 C6Z1WI 44449555 Ki = 127 nM T92072 C62URD 44449567 Ki = 990 nM T92072 CO8P4M 44449568 Ki = 1588 nM T92072 CO04QJ 44449570 Ki = 5513 nM T92072 C9ZH1F 44449591 Ki = 1856 nM T92072 CI80QT 44449598 Ki = 5768 nM T92072 C19JVY 44449599 Ki = 1095 nM T92072 CZ95HM 44449626 Ki = 4960 nM T92072 C9OU7X 44449633 Ki = 868 nM T92072 C0PO3H 44449634 Ki = 3467 nM T92072 CZUB58 44449635 Ki = 366 nM T92072 C80YCR 44449636 Ki = 2197 nM T92072 C0LAZ6 44449655 Ki = 7628 nM T92072 CRES01 44449665 Ki = 568 nM T92072 C9ODF3 44449666 Ki = 375 nM T92072 C74VPR 44449668 Ki = 1255 nM T92072 C5X0UL 44449693 Ki = 6470 nM T92072 CXK0M2 44449706 Ki = 5525 nM T92072 C1DLR5 44449707 Ki = 4938 nM T92072 C0HZ1F 44449728 Ki = 1938 nM T92072 CLGN80 44449740 Ki = 401 nM T92072 C6SMZ7 44449742 Ki = 1963 nM T92072 C9KA4M 44449744 Ki = 1590 nM T92072 C95SAB 44449745 Ki = 813 nM T92072 C3N9OC 44449746 Ki > 100000 nM T92072 CP78RA 44450158 Ki = 316 nM T92072 C0E3MF 44450161 Ki = 471 nM T92072 C6I3MS 44450188 Ki = 17514 nM T92072 C0SU7H 44450189 Ki = 4475 nM T92072 C8W5YK 44450190 Ki = 14454 nM T92072 CHP5W0 44450290 Ki = 0.67 nM T92072 CCMZ32 44450517 Ki = 314 nM T92072 C6VFH5 44450829 Ki = 363.08 nM T92072 C76MCE 44450982 Ki = 676.08 nM T92072 C6PK0V 44450983 Ki = 43 nM T92072 CN7TA8 44451127 Ki = 89.13 nM T92072 C75LZM 44451224 Ki = 269.15 nM T92072 C50QVJ 44451283 Ki = 501.19 nM T92072 CEL5J8 44451482 Ki = 537.03 nM T92072 CYOF07 44451499 Ki = 13 nM T92072 CO0UD1 44451500 Ki = 6.8 nM T92072 CGS85Y 44451501 Ki = 27.9 nM T92072 CL8PQ6 44451524 Ki = 17.3 nM T92072 C3VZR4 44451525 Ki = 6.4 nM T92072 C1T8VP 44451582 Ki = 2.9 nM T92072 C8JOS1 44451604 Ki = 15.6 nM T92072 CN7KU2 44451658 Ki = 115 nM T92072 CG1FV5 44451682 Ki = 102 nM T92072 C0JB2Q 44451683 Ki = 8.3 nM T92072 C4J3XI 44451738 Ki = 2.8 nM T92072 C8GL3J 44451787 Ki = 27.9 nM T92072 C8M6EA 44451790 Ki = 1.8 nM T92072 COVW35 44451815 Ki = 12.6 nM T92072 C3UIY5 44451817 Ki = 92.3 nM T92072 CA76ZH 44451846 Ki = 5.3 nM T92072 C4O5SM 44451848 Ki = 17.6 nM T92072 C1DVS2 44451849 Ki = 9.4 nM T92072 CG3F6S 44451878 Ki = 18.4 nM T92072 C3MEY2 44451881 Ki = 43 nM T92072 CUO7F6 44451902 Ki = 13.4 nM T92072 CDP23H 44451903 Ki = 2.9 nM T92072 CP26ZR 44451904 Ki = 8.1 nM T92072 C4A3TB 44451923 Ki = 5.7 nM T92072 CT0IR5 44452381 IC50 = 4279 nM T92072 CS3T6Y 44452401 IC50 = 605 nM T92072 CN0BP8 44452405 Ki = 102.33 nM T92072 C4APQ6 44452407 Ki = 45.71 nM T92072 CAO9T8 44452429 IC50 = 4950 nM T92072 C1KXG7 44452431 Ki = 199.53 nM T92072 C6AG2Y 44452434 Ki = 63.1 nM T92072 CJW91V 44452435 Ki = 12.59 nM T92072 CX3EL6 44452450 IC50 = 867 nM T92072 C87QHW 44452454 Ki = 537.03 nM T92072 C0PER5 44452455 Ki = 112.2 nM T92072 CB0S6P 44452475 Ki = 3715.35 nM T92072 C3G5HY 44452478 Ki = 331.13 nM T92072 CXP3W0 44452488 IC50 = 351 nM T92072 C6NZC5 44452489 IC50 = 12 nM T92072 CTC57Y 44452490 Ki = 58.88 nM T92072 C8WO7J 44452491 Ki = 575.44 nM T92072 CTMF29 44452493 Ki = 134.9 nM T92072 C9MIL8 44452508 IC50 = 0.9 nM T92072 CH3RM7 44452509 IC50 = 48 nM T92072 C6DU3Q 44452514 Ki = 74.13 nM T92072 CG74SF 44452515 Ki = 302 nM T92072 CDU2I1 44452516 Ki = 141.25 nM T92072 CU24GW 44452530 IC50 = 0.3 nM T92072 CRL81W 44452532 IC50 = 21 nM T92072 C2K9ME 44452533 IC50 = 15 nM T92072 C18BXC 44452535 Ki = 3.162 nM T92072 CWF9E6 44452536 Ki = 3.981 nM T92072 CSFV93 44452539 Ki = 93.33 nM T92072 C8U4PX 44452562 IC50 = 0.12 nM T92072 C9A7NE 44452564 IC50 = 28 nM T92072 CZEV82 44452582 IC50 = 68 nM T92072 C2JBG6 44452604 IC50 = 224 nM T92072 CN1JQ8 44452606 IC50 = 2.6 nM T92072 CIJ24N 44452625 IC50 = 7 nM T92072 CY1FO3 44452673 IC50 = 710 nM T92072 CPLM63 44452690 IC50 = 410 nM T92072 C8SIX2 44452695 Ki = 33.11 nM T92072 C4B7VM 44454763 IC50 >= 10000 nM T92072 C2EQM1 44454764 IC50 >= 10000 nM T92072 CWZG75 44454788 IC50 >= 10000 nM T92072 C9YD4Q 44454789 IC50 >= 10000 nM T92072 CN7Y2F 44454816 IC50 >= 10000 nM T92072 CTWR48 44454817 IC50 >= 10000 nM T92072 CU5XL2 44454818 IC50 >= 10000 nM T92072 CB67EY 44454849 Ki = 237 nM T92072 C60CIT 44454850 IC50 >= 10000 nM T92072 CZU8C6 44454851 IC50 >= 10000 nM T92072 CH5SW9 44454853 Ki = 345 nM T92072 CL39AN 44454883 Ki = 404 nM T92072 C7UK9H 44454885 IC50 >= 10000 nM T92072 C52HBA 44454886 IC50 >= 10000 nM T92072 C7APO0 44454922 IC50 >= 10000 nM T92072 C52LGN 44454923 IC50 >= 10000 nM T92072 C6CO9J 44454925 IC50 >= 10000 nM T92072 CXOS03 44457466 Ki = 13500 nM T92072 C6A9OT 44457469 Ki = 11700 nM T92072 CS1F5E 44457473 Ki = 379 nM T92072 CR58PU 44457922 Ki = 3599 nM T92072 CIDT05 44457923 Ki = 1793 nM T92072 C0GTF5 44457953 Ki = 9533 nM T92072 C2GTV4 44458220 Ki = 60 nM T92072 C4DL5C 44469677 IC50 > 10000 nM T92072 C2T8CA 44520931 Ki = 41 nM T92072 CT8OY0 44520932 Ki = 105 nM T92072 CXU2F8 44520933 Ki = 103 nM T92072 C5V6OI 44520934 Ki = 202 nM T92072 CKC3Q4 44520935 Ki = 223 nM T92072 C6H7PM 44520936 Ki = 409 nM T92072 CLCB53 44520937 Ki = 586 nM T92072 CD29LZ 44520938 Ki = 1112 nM T92072 CI82SB 44520939 Ki = 595 nM T92072 CC97FL 44520940 Ki = 921 nM T92072 CB7K2Y 44520941 Ki = 222 nM T92072 CL3NH5 44520942 Ki = 66 nM T92072 CU3GW7 44520943 Ki = 48 nM T92072 C6CEV4 44520944 Ki = 38 nM T92072 CD9Q7Z 44520945 Ki = 408 nM T92072 CCS87V 44520946 Ki = 40 nM T92072 C21CFR 44520947 Ki = 1377 nM T92072 C6HN5S 44520948 Ki = 67 nM T92072 C8DZR0 44520949 Ki = 118 nM T92072 CH7FI4 44520950 Ki = 1242 nM T92072 CO82QN 44520951 Ki = 252 nM T92072 CGH3X0 44520952 Ki = 478 nM T92072 CJ4NA8 44520953 Ki > 10000 nM T92072 C49KZA 44520954 Ki = 9171 nM T92072 CW76RP 44520955 Ki = 1670 nM T92072 CQK20C 44520956 Ki > 10000 nM T92072 C6KJC7 44520957 Ki = 38 nM T92072 CIR5M0 44520958 Ki = 31 nM T92072 CMU48O 44520959 Ki = 394 nM T92072 C5L2GJ 44520960 Ki = 56 nM T92072 CN0MR1 44520961 Ki = 94 nM T92072 C7AGL5 44520962 Ki = 83 nM T92072 CWV6A8 44520963 Ki = 720 nM T92072 CWR28D 44520964 Ki = 199 nM T92072 C9HO8N 44520965 Ki = 276 nM T92072 C4RDH8 44520966 Ki > 10000 nM T92072 C38PAD 44520967 Ki = 7902 nM T92072 C5QPO3 44520968 Ki = 1157 nM T92072 CZ4I9A 44520969 Ki = 395 nM T92072 C8Y4MD 44520970 Ki > 10000 nM T92072 CZ37SW 44520971 Ki = 314 nM T92072 CZO52W 44520972 Ki = 435 nM T92072 CK69IO 44520973 Ki = 576 nM T92072 CEP2L4 44520974 Ki = 504 nM T92072 CJ97HI 44520975 Ki = 2545 nM T92072 CZ6F9S 44520976 Ki = 133 nM T92072 C4Q5JZ 44520977 Ki = 77.5 nM T92072 CX54QG 44520978 Ki = 57 nM T92072 C9EH4F 44520979 Ki = 89 nM T92072 CQ71XC 44520980 Ki = 172 nM T92072 CEO4P7 44520981 Ki = 270 nM T92072 C31SUP 44520982 Ki = 368 nM T92072 CNR53B 44520983 Ki = 385 nM T92072 C3ZCH7 44520984 Ki = 277 nM T92072 C3MZC5 44520985 Ki = 270 nM T92072 C7HVU4 44520987 Ki = 90 nM T92072 C5M3GT 44520988 Ki = 38 nM T92072 CJ57RW 44537897 Ki = 48.2 nM T92072 CLI7K5 44562753 Ki = 500 nM T92072 CVW3N2 44563977 Ki = 120 nM T92072 C4LI1U 44564568 Ki = 1833 nM T92072 C4VJB3 44564569 Ki = 10000 nM T92072 CJ94UT 44564881 Ki = 402 nM T92072 C75ZAH 44564883 Ki = 447 nM T92072 CI9BH4 44564926 Ki = 599 nM T92072 CPF51G 44564927 Ki = 1847 nM T92072 CD0W8R 44564928 Ki = 3237 nM T92072 CUX0Q7 44564978 Ki > 10000 nM T92072 CL72ZU 44564979 Ki = 564 nM T92072 CP2FL0 44564980 Ki = 201 nM T92072 CO1Z3J 44564981 Ki = 2850 nM T92072 CIEH58 44565032 Ki = 330 nM T92072 CTYJ67 44565076 Ki = 1265 nM T92072 C9WV1X 44565077 Ki = 1110 nM T92072 C65ZWP 44565078 Ki = 1053 nM T92072 CO1RK2 44565079 Ki = 616 nM T92072 C5C3RG 44565133 Ki = 2972 nM T92072 CA5B6M 44565134 Ki = 1473 nM T92072 CFJ6D2 44565135 Ki = 1056 nM T92072 C1LK8I 44565136 Ki = 1072 nM T92072 C2B3MD 44565183 Ki = 1211 nM T92072 C6TXF8 44565184 Ki = 1191 nM T92072 CV6I0P 44567439 Ki > 100000 nM T92072 C2RJ7Q 44568838 Ki = 17.3 nM T92072 CW0B5D 44570367 Ki > 1000 nM T92072 C9BA3H 44570369 Ki > 1000 nM T92072 C24CRG 44570413 Ki > 1000 nM T92072 C6EAT9 44570414 Ki > 1000 nM T92072 CTS6P4 44570415 Ki > 1000 nM T92072 CP93SE 44570416 Ki > 1000 nM T92072 C6NJP3 44570454 Ki > 1000 nM T92072 CC6TW2 44570455 Ki > 1000 nM T92072 CG9BR2 44570456 Ki > 1000 nM T92072 C9FV0G 44570457 Ki > 1000 nM T92072 CC51RV 44570458 Ki > 1000 nM T92072 CSMN18 44570493 Ki > 1000 nM T92072 CMD87Q 44572294 Ki > 100000 nM T92072 CSL0G8 44572353 Ki > 100000 nM T92072 C0ETQ1 44572354 Ki > 100000 nM T92072 C7D2GC 44572410 Ki > 100000 nM T92072 C9VS8P 44572470 Ki > 100000 nM T92072 CDZ14G 44572472 Ki > 100000 nM T92072 C8Y0EI 44574117 Ki = 2.2 nM T92072 CZDG39 44574118 Ki = 17.8 nM T92072 CZX7N5 44574165 Ki = 10 nM T92072 CUH78B 44574194 Ki = 20.4 nM T92072 CMFB42 44574222 Ki = 0.4 nM T92072 CA31JY 44579667 Ki = 1600 nM T92072 CR0GX1 44579668 Ki = 870 nM T92072 C7RA4N 44579669 Ki = 252 nM T92072 C2TZQ6 44579670 Ki = 4820 nM T92072 CZS2C8 44579671 Ki = 1010 nM T92072 CCN45J 44579672 Ki = 6630 nM T92072 CF04WK 44579673 Ki = 3000 nM T92072 CRS81G 44579674 Ki = 1110 nM T92072 CF2O3K 44579675 Ki = 1790 nM T92072 CL18FO 44579714 Ki = 3040 nM T92072 C5TKU6 44579715 Ki = 1600 nM T92072 CI4FW1 44579716 Ki = 1760 nM T92072 CZ7NV2 44579717 Ki = 1120 nM T92072 CHC02W 44581364 Ki = 3580 nM T92072 C0X4UM 44581365 Ki = 1280 nM T92072 CHR9Z1 44581366 Ki = 6780 nM T92072 CB1Q8U 44581367 Ki = 3970 nM T92072 CINU98 44581368 Ki = 2420 nM T92072 CMB71E 44581369 Ki = 1240 nM T92072 C27QRK 44581397 Ki = 3710 nM T92072 CS8QR0 44581398 Ki = 3500 nM T92072 C9S3YK 44581428 Ki > 6700 nM T92072 CDT8Z2 44581429 Ki = 6300 nM T92072 CWBF57 44581430 Ki > 10000 nM T92072 C8ZU0M 44581431 Ki = 9460 nM T92072 C60UGT 44581432 Ki = 3420 nM T92072 C7CAH0 44581471 Ki > 10000 nM T92072 C76WPB 44581472 Ki > 10000 nM T92072 CZ72WU 44581866 Ki = 222 nM T92072 C8FEZ9 44581894 Ki = 1533 nM T92072 CM6AK4 44581895 Ki = 4695 nM T92072 C6EUC0 44581896 Ki = 1640 nM T92072 CCB34Q 44582614 Ki = 1.61 nM T92072 CSM58E 44582652 Ki = 9.13 nM T92072 CA5R4M 44582653 Ki = 9.16 nM T92072 CR95SV 44582654 Ki = 64.7 nM T92072 C8G4TH 44582690 Ki = 1060 nM T92072 CV5F9X 44582691 Ki = 2970 nM T92072 C71SDJ 44582723 Ki = 250 nM T92072 CLW60K 44582724 Ki = 4.09 nM T92072 CH07JS 44582725 Ki = 6.96 nM T92072 CZ91EO 44582726 Ki = 0.71 nM T92072 C9Y8VU 44583006 Ki > 10000 nM T92072 CR3LW0 44583035 Ki = 79 nM T92072 C7D9YB 44586199 Ki = 2700 nM T92072 CY2MH0 44586253 Ki = 12.3 nM T92072 CY03KI 44586254 Ki = 4215 nM T92072 CC7FH5 44586717 Ki = 779 nM T92072 C7S1MY 44586718 Ki = 2379 nM T92072 C6IO7C 44587956 Ki = 79 nM T92072 CUG8E4 44587957 Ki = 224 nM T92072 C6IE2F 44588394 Ki = 25 nM T92072 CG1JD0 44588395 Ki = 83 nM T92072 CBL10K 44588516 Ki = 63 nM T92072 C0UD5O 44588517 Ki = 240 nM T92072 CVW37M 44597868 Ki = 1600 nM T92072 CV4TA7 44597869 Ki = 839 nM T92072 C5KTS9 44597870 Ki = 513 nM T92072 CUO03D 44597871 Ki = 109 nM T92072 C5ZLC3 44598835 Ki = 5310 nM T92072 C6LXZ8 44598836 Ki = 8740 nM T92072 CFIA83 44631910 IC50 = 0.6 nM T92072 CDTA58 45136848 Ki = 129 nM T92072 C36SXK 45136852 Ki = 150 nM T92072 CKZE75 45258867 IC50 = 933.25 nM T92072 C0ZU9Y 45258869 IC50 = 229.09 nM T92072 C37HPT 45258970 IC50 = 83.18 nM T92072 CLB20G 45266415 Ki > 100000 nM T92072 CU84YS 45266426 Ki > 100000 nM T92072 CNO3D6 45267119 Ki = 2004 nM T92072 C1I6ZN 45267125 Ki = 140 nM T92072 C6BDH1 45267130 Ki = 157 nM T92072 CHK6Z9 45267243 Ki = 1060 nM T92072 CJZ29E 45267454 Ki = 1410 nM T92072 C24KLI 45267987 Ki = 58 nM T92072 CG7M5U 45267990 Ki = 72 nM T92072 CSGE26 45268313 Ki = 921 nM T92072 CSP4L8 45268863 Ki = 298 nM T92072 C1IL3E 45268869 Ki = 12.2 nM T92072 C7EL9J 45269703 Ki = 311 nM T92072 C57YDT 45269835 Ki = 795 nM T92072 C0Q7RF 45269838 Ki = 2480 nM T92072 CW8U6A 45270537 Ki = 770 nM T92072 CJP69G 45270541 Ki = 39 nM T92072 CX78GF 45271359 Ki = 2062 nM T92072 CY3A1D 45271366 Ki = 80 nM T92072 C20RJQ 45271709 Ki = 132 nM T92072 CK1H3O 45272255 Ki = 3540 nM T92072 CZ3D2A 45272256 Ki = 884 nM T92072 C6O8XQ 45273122 Ki = 102 nM T92072 C5SRP3 45274224 Ki > 1000 nM T92072 CAM9S8 45274225 Ki = 618 nM T92072 CWZV56 45274227 Ki = 283 nM T92072 C9MB3Z 45274228 Ki = 263 nM T92072 C19YWV 45274324 Ki = 91 nM T92072 CV4R3I 45274328 Ki = 49.6 nM T92072 C5OBS2 45274330 Ki = 26.1 nM T92072 CU4XV8 45274426 Ki = 516 nM T92072 CS3CF1 45274431 Ki = 2998 nM T92072 CBX3M6 45275056 Ki = 222 nM T92072 CBUV31 45275058 Ki = 151 nM T92072 C6TC5O 45275060 Ki > 1000 nM T92072 CE7F8G 45275061 Ki > 610 nM T92072 CSEL27 45275170 Ki = 1772 nM T92072 CYL7Z2 45275171 Ki > 1000 nM T92072 CUMC92 45275172 Ki = 266 nM T92072 CV7L4T 45275173 Ki = 123 nM T92072 C8LB2S 45275287 Ki = 24.8 nM T92072 COVY03 45275517 Ki = 298 nM T92072 CX49ZH 45275619 Ki = 223 nM T92072 CCL28P 45275713 Ki > 610 nM T92072 CK2G4Y 45275714 Ki > 594 nM T92072 C4ZT2C 45275715 Ki = 122 nM T92072 CTN65H 45275716 Ki = 1418 nM T92072 CP82KG 45275717 Ki = 1491 nM T92072 CQC5T8 45275718 Ki = 186 nM T92072 CU8HY4 45275719 Ki = 439 nM T92072 CLE92Q 45275818 Ki = 1416 nM T92072 C8P0ZA 45275819 Ki = 3163 nM T92072 CQL3P8 45275820 Ki = 2332 nM T92072 C6BIV9 45275821 Ki = 106 nM T92072 CX5F0H 45275823 Ki = 2784 nM T92072 C8DPZ0 45275824 Ki = 861 nM T92072 CO2E5P 45278533 Ki = 290 nM T92072 C3WGV4 45278535 Ki = 630 nM T92072 CJED13 45278537 Ki = 620 nM T92072 CC4XE8 45278538 Ki = 840 nM T92072 CIV2G3 45278539 Ki = 1630 nM T92072 CQYO92 45278617 Ki = 2070 nM T92072 C1GP7V 45278618 Ki = 130 nM T92072 C6WVU9 45278619 Ki = 8430 nM T92072 CNG16P 45278621 Ki = 210 nM T92072 CQ5J7L 45278622 Ki = 3895 nM T92072 C15LZX 45278623 Ki = 2964 nM T92072 C93ZXP 45278697 Ki = 3220 nM T92072 CHL5W1 45278699 Ki = 5050 nM T92072 C9V6XY 45278700 Ki = 1010 nM T92072 CMJ06I 45278701 Ki = 3250 nM T92072 CD7GE2 45278783 Ki = 2950 nM T92072 CVDZ38 45278784 Ki = 980 nM T92072 CUE83H 45278785 Ki = 2990 nM T92072 CVDJ21 45278787 Ki = 1810 nM T92072 CXU4S7 45278863 Ki = 2350 nM T92072 CKVQ57 45278864 Ki = 1080 nM T92072 CG23WV 45278865 Ki = 710 nM T92072 CZI7V5 45278866 Ki = 1420 nM T92072 CJ5G3X 45278867 Ki = 1240 nM T92072 CJ1MA9 45278868 Ki = 190 nM T92072 CX4B6U 45278944 Ki = 780 nM T92072 C5S6IP 45278946 Ki = 1670 nM T92072 C3LI4D 45278947 Ki = 2100 nM T92072 CZ7T1U 45278948 Ki = 730 nM T92072 C96HNR 45278949 Ki = 2700 nM T92072 CIC9V4 45279186 Ki = 188 nM T92072 CZ42MB 45279272 Ki = 640 nM T92072 CG6N9M 45279273 Ki = 245 nM T92072 C85DGX 45279274 Ki = 725 nM T92072 CXZ01P 45279275 Ki > 610 nM T92072 CJB9L4 45279276 Ki = 300 nM T92072 CV29MU 45279277 Ki = 140 nM T92072 CES35K 45279356 Ki = 190 nM T92072 C45JDQ 45279358 Ki > 930 nM T92072 CT4LX5 45279360 Ki = 680 nM T92072 C9PV1L 45279361 Ki = 1070 nM T92072 CQ7U1I 45279362 Ki = 500 nM T92072 CJL90G 45279445 Ki = 40.2 nM T92072 CU6P4F 45279446 Ki > 600 nM T92072 CQ4WL3 45279448 Ki > 1100 nM T92072 CR73ZU 45279449 Ki = 460 nM T92072 CMH6F3 45279451 Ki = 2730 nM T92072 C64KIA 45279539 Ki = 1020 nM T92072 CIZS47 45279541 Ki = 6430 nM T92072 CJ53BU 45279542 Ki = 1890 nM T92072 CN8TV0 45279543 Ki > 10000 nM T92072 C1O0IT 45279544 Ki = 2130 nM T92072 CP47WG 45279545 Ki = 2480 nM T92072 C0C1LT 45279632 Ki = 610 nM T92072 CR07AK 45279633 Ki = 710 nM T92072 C15ZWH 45279636 Ki = 1050 nM T92072 CQCA71 45279637 Ki = 620 nM T92072 CLEA65 45279724 Ki = 3320 nM T92072 C6S0WZ 45279725 Ki = 1680 nM T92072 C1H4CQ 45279727 Ki = 100 nM T92072 CP74GQ 45279728 Ki = 2720 nM T92072 CY8R1U 45279729 Ki = 3550 nM T92072 C6ZLX7 45279730 Ki = 2300 nM T92072 C6MR2P 45279822 Ki = 790 nM T92072 CH52XG 45279823 Ki = 2890 nM T92072 C86KCE 45279824 Ki = 1340 nM T92072 CFV13P 45279825 Ki = 4000 nM T92072 C5B7LP 45279828 Ki = 2230 nM T92072 CPG3L9 45481619 Ki = 13.7 nM T92072 C2ZI4P 45481621 Ki = 129 nM T92072 CCMX92 45481749 Ki = 185 nM T92072 CXM9F4 45481750 Ki = 139 nM T92072 CBOG84 45481751 Ki = 1460 nM T92072 CLZV08 45481752 Ki = 441 nM T92072 C3MPR1 45481753 Ki = 410 nM T92072 CB52VK 45481754 Ki = 80.2 nM T92072 C5W4NR 45481755 Ki = 18.5 nM T92072 CQOB79 45481756 Ki = 154 nM T92072 CB8NA2 45481757 Ki = 148 nM T92072 CL68UB 45481758 Ki = 461 nM T92072 CY2WO6 45481759 Ki = 84.3 nM T92072 CV43FT 45481760 Ki = 115 nM T92072 C50HVN 45481761 Ki = 84.3 nM T92072 C4C0QV 45481762 Ki = 622 nM T92072 C16LEJ 45481763 Ki = 1850 nM T92072 C1TB7C 45481764 Ki = 22.8 nM T92072 CP02LD 45481765 Ki = 596 nM T92072 C0L9GH 45481766 Ki = 557 nM T92072 CH54CA 45481767 Ki = 133 nM T92072 C7GF4H 45481768 Ki = 140 nM T92072 C1FA8U 45481769 Ki = 190 nM T92072 C2TWL7 45481770 Ki = 57.5 nM T92072 C5H7SZ 45481771 Ki = 381 nM T92072 C12JUY 45482074 Ki = 605 nM T92072 C0FG6J 45482075 Ki = 388 nM T92072 CQ5ZF6 45482076 Ki = 741 nM T92072 CMI3P8 45482077 Ki = 726 nM T92072 CDSG82 45482078 Ki = 307 nM T92072 C01FXN 45482079 Ki = 256 nM T92072 CE3TD2 45482080 Ki = 160 nM T92072 C0IT6Y 45482081 Ki = 121 nM T92072 C0RN6K 45482082 Ki = 170 nM T92072 CD6I4G 45482083 Ki = 768 nM T92072 CZ30JX 45482084 Ki = 241 nM T92072 CY49LO 45482085 Ki = 70.1 nM T92072 C1VEW8 45482086 Ki = 25.5 nM T92072 C8Q6KD 45482087 Ki = 908 nM T92072 CP5LN6 45482088 Ki = 963 nM T92072 C12UZF 45482089 Ki = 71.1 nM T92072 CIF06H 45482090 Ki = 22.6 nM T92072 CDK76E 45482091 Ki = 786 nM T92072 CC52GU 45482092 Ki = 1170 nM T92072 CL39ZH 45482093 Ki = 872 nM T92072 C8PQ9W 45482094 Ki = 13.2 nM T92072 COL2R3 45482462 Ki = 444 nM T92072 CNDA49 45482464 Ki = 51.8 nM T92072 CS2D7I 45482869 Ki = 800 nM T92072 C8JMG7 45482870 Ki = 53800 nM T92072 C64KXS 45482874 Ki = 10200 nM T92072 CH4O5W 45483954 Ki = 700 nM T92072 C76YLH 45483955 Ki = 260 nM T92072 CNP07M 45483958 Ki = 482 nM T92072 C8PFI3 45483960 Ki = 2320 nM T92072 CXP5T3 45483961 Ki = 454 nM T92072 C1LM8Y 45486932 Ki = 8730 nM T92072 CPCD97 46175652 IC50 = 16 nM T92072 CD30NG 46175736 IC50 = 5.1 nM T92072 C8GLI6 46175737 IC50 = 8 nM T92072 C15UPZ 46175738 IC50 = 7.3 nM T92072 CQRB27 46175914 IC50 = 277 nM T92072 CQ9NB4 46176000 IC50 = 6.4 nM T92072 C28AUS 46202865 Ki = 467.74 nM T92072 CH0TL3 46203191 Ki = 245.47 nM T92072 C05ORG 46203192 Ki = 309.03 nM T92072 C1SNV5 46203193 EC50 = 51.29 nM T92072 CZ0H6L 46203194 Ki = 275.42 nM T92072 C96EWH 46203499 Ki = 346.74 nM T92072 CDE9K0 46203500 Ki = 457.09 nM T92072 CJW69T 46203822 Ki = 1258.93 nM T92072 C5FME6 46204157 EC50 = 8500 nM T92072 CE72PC 46204158 EC50 = 3700 nM T92072 CEKW03 46204482 EC50 = 5200 nM T92072 CRE07N 46205479 Ki = 339 nM T92072 C5CV8H 46205480 Ki = 1010 nM T92072 C5GM2E 46205481 Ki = 4860 nM T92072 C7YD4H 46205482 Ki = 2890 nM T92072 C1MS4I 46205483 Ki = 9730 nM T92072 CG60ME 46205484 Ki > 300000 nM T92072 C4B5NU 46205485 Ki = 121 nM T92072 CQK0G9 46205805 Ki = 1570 nM T92072 CLW1U9 46205806 Ki = 39.1 nM T92072 CRS91E 46205807 Ki = 204 nM T92072 CT8E0B 46205808 Ki = 498 nM T92072 C5EZ8J 46205809 Ki = 289 nM T92072 CS3MD6 46205810 Ki = 622 nM T92072 CLAP45 46206128 Ki = 2530 nM T92072 CK85FB 46206129 Ki > 30000 nM T92072 CTZ2J4 46206130 Ki > 30000 nM T92072 CV1HG3 46206131 Ki > 30000 nM T92072 C0XJ1G 46206132 Ki > 30000 nM T92072 CT4C0Q 46206133 Ki > 10000 nM T92072 C9TY8Z 46206464 Ki > 10000 nM T92072 COIG13 46206465 Ki = 313 nM T92072 C5NGI1 46206466 Ki = 270 nM T92072 CYZ9G2 46206467 Ki = 562 nM T92072 C8JDB5 46206468 Ki = 2290 nM T92072 C45TYC 46206469 Ki = 4850 nM T92072 CHO5B4 46206809 Ki = 24400 nM T92072 CDS62V 46206810 Ki > 30000 nM T92072 C7RP3G 46206811 Ki = 23200 nM T92072 CMIE96 46213946 IC50 = 2 nM T92072 C5Q3GH 46225677 Ki = 74 nM T92072 C9X6TQ 46225735 Ki = 72.5 nM T92072 CH34QJ 46226779 Ki = 69.5 nM T92072 C1FO0X 46226780 Ki = 4.83 nM T92072 COZQ07 46226791 Ki = 6.58 nM T92072 CGH6A8 46226792 Ki = 33.1 nM T92072 C3GC7Q 46226793 Ki = 6.27 nM T92072 CZ4Y1T 46226797 Ki = 48.6 nM T92072 C5TUH7 46226812 Ki = 5.4 nM T92072 C25QHA 46226822 Ki = 9.27 nM T92072 CSR2C5 46226840 Ki = 159 nM T92072 C01JNB 46226841 Ki = 23.6 nM T92072 C8GIE9 46226873 Ki = 4070 nM T92072 CF9E0O 46227337 EC50 = 13200 nM T92072 C7XO8T 46227350 EC50 = 11500 nM T92072 CBG2X7 46227370 EC50 = 7200 nM T92072 CN5EP8 46227373 EC50 = 9100 nM T92072 C2M8NA 46227374 EC50 = 7900 nM T92072 C50EON 46227379 EC50 = 12100 nM T92072 CV9EU1 46227384 EC50 = 13100 nM T92072 C9KXU7 46227386 EC50 > 20000 nM T92072 CWY1C9 46227392 EC50 = 15500 nM T92072 CIV90Y 46227394 EC50 = 8900 nM T92072 CN7QW2 46227402 EC50 = 7800 nM T92072 C5C0LN 46228971 Ki = 57.4 nM T92072 CHTV64 46229143 Ki = 23.2 nM T92072 CJ8CU7 46229272 Ki = 0.58 nM T92072 C1KVY2 46230151 EC50 > 10000 nM T92072 CV45DT 46230237 EC50 > 10000 nM T92072 C7EWV0 46230238 EC50 > 10000 nM T92072 CT4AE8 46230239 EC50 > 10000 nM T92072 C21NRT 46230240 EC50 > 10000 nM T92072 C1B9ZU 46230246 EC50 > 10000 nM T92072 C80CWB 46230290 EC50 = 4100 nM T92072 CM1H7R 46233161 Ki = 93.33 nM T92072 CI1Z4R 46233211 Ki = 223.87 nM T92072 CW54HP 46233214 Ki = 147.91 nM T92072 C4HE1X 46233278 Ki = 218.78 nM T92072 CT5CF9 46233315 Ki = 676.08 nM T92072 CV27IG 46233316 Ki = 407.38 nM T92072 C8GM6X 46233347 Ki = 389.05 nM T92072 C17TOR 46233377 Ki = 95.5 nM T92072 C3MCA6 46233378 Ki = 100 nM T92072 C8PJ7D 46233379 Ki = 120.23 nM T92072 C7LY3J 46233380 Ki = 194.98 nM T92072 C48HIY 46233446 Ki = 93.33 nM T92072 CEXP72 46237805 Ki = 584.7 nM T92072 C5TRP3 46237926 Ki = 312 nM T92072 C9GM2W 46237927 Ki = 2500 nM T92072 CG57HC 46237928 Ki = 334 nM T92072 C0Z1AL 46237929 Ki = 1037 nM T92072 CCJ09W 46237930 Ki = 1081.6 nM T92072 CN36TB 46237931 Ki > 10000 nM T92072 C7US4A 46237932 Ki > 10000 nM T92072 CX5RZ3 46238063 Ki > 10000 nM T92072 CB6P5J 46238064 Ki = 53 nM T92072 C5LKY8 46238065 Ki > 10000 nM T92072 CM6K9V 46238066 Ki > 10000 nM T92072 CMD67R 46238067 Ki = 290 nM T92072 C9S4VL 46238068 Ki > 10000 nM T92072 C7DPI4 46238208 Ki > 10000 nM T92072 CP9QS1 46238209 Ki = 27 nM T92072 CI3S2V 46238210 Ki = 2400 nM T92072 CS4T7D 46238211 Ki = 1050 nM T92072 CD60TM 46238212 Ki = 1700 nM T92072 CX6OK2 46238213 Ki > 10000 nM T92072 CAY7J1 46238338 Ki > 10000 nM T92072 C6PQR8 46238339 Ki > 10000 nM T92072 CWS95Q 46238340 Ki > 10000 nM T92072 CW41JP 46238341 Ki > 10000 nM T92072 CO5J9W 46238636 IC50 = 10 nM T92072 CES60L 46238684 IC50 = 15 nM T92072 C5H9JS 46238686 IC50 = 6 nM T92072 CXI4A9 46238694 IC50 = 11 nM T92072 C0I1XV 46238729 IC50 = 87 nM T92072 C3L9OR 46240228 IC50 = 13 nM T92072 C28NVK 46257086 Ki = 19498.45 nM T92072 C9O2KM 46391804 Ki = 512.86 nM T92072 CKGM09 46837704 Ki = 75.86 nM T92072 CRG03C 46837705 Ki = 1.738 nM T92072 C71GBF 46861670 Ki = 245 nM T92072 CYC93U 46861671 Ki = 26.2 nM T92072 CLH9D6 46861672 Ki = 105 nM T92072 C9GCO1 46861768 Ki = 32.9 nM T92072 C9X2WT 46861769 Ki = 116 nM T92072 C0RFZ6 46861770 Ki = 85 nM T92072 CDCK67 46861780 Ki = 32.7 nM T92072 CK8D9S 46861781 Ki = 35.6 nM T92072 CIB5U2 46861782 Ki = 256 nM T92072 CC50RJ 46863665 Ki = 17 nM T92072 CU09WX 46865328 Ki = 228.4 nM T92072 CB62WH 46865329 Ki = 147.9 nM T92072 CHY8V9 46865434 Ki = 19.01 nM T92072 C5QXL9 46866591 Ki = 82 nM T92072 C8VJ9K 46866592 Ki = 931 nM T92072 CK9AU5 46866593 Ki = 374 nM T92072 CA2S6O 46875997 Ki = 1176 nM T92072 CC5OH2 46876751 Ki = 325 nM T92072 C2JQ9I 46876986 EC50 = 9.2 nM T92072 C95MDF 46876987 EC50 = 21.5 nM T92072 CC7B4U 46877219 Ki = 750 nM T92072 CY6S3U 46877262 Ki = 240 nM T92072 CT82OL 46877263 Ki = 730 nM T92072 CKUF93 46877269 Ki = 725 nM T92072 CLU0A9 46877270 Ki = 280 nM T92072 C5D2NU 46877277 Ki = 415 nM T92072 CCH83Y 46877278 Ki = 445 nM T92072 CP3RO7 46877284 Ki = 250 nM T92072 CHI72K 46877285 Ki = 350 nM T92072 C3FJZ9 46877286 Ki = 300 nM T92072 CWD63T 46877289 Ki = 206 nM T92072 COJW51 46877298 Ki = 350 nM T92072 C5MB9D 46877311 Ki = 290 nM T92072 CJ6LH9 46877313 Ki = 250 nM T92072 CFV06U 46877320 Ki = 280 nM T92072 C8H2FW 46877321 Ki = 250 nM T92072 C8C6VB 46877325 Ki = 380 nM T92072 C3F5EW 46877333 Ki = 700 nM T92072 CNYJ02 46877335 Ki = 350 nM T92072 C50XUB 46880372 Ki = 285 nM T92072 CZJ2V5 46880373 Ki = 289 nM T92072 CL8UH3 46880375 Ki = 250 nM T92072 CQ93IM 46880419 Ki = 25 nM T92072 CMCX40 46880420 Ki = 914 nM T92072 C7P6TS 46880421 Ki = 320 nM T92072 CKB31F 46880422 Ki = 702 nM T92072 CH5B6C 46880424 Ki = 1727 nM T92072 CB9TI2 46880470 Ki = 635 nM T92072 COQ7X3 46880474 Ki = 123 nM T92072 C2SM9Q 46880475 Ki = 14 nM T92072 CV10FQ 46880506 Ki = 58 nM T92072 CMP72U 46880507 Ki = 35 nM T92072 CM36IE 46880508 Ki = 940 nM T92072 C61JDB 46880510 Ki = 338 nM T92072 CGZ31A 46885889 Ki = 0.096 nM T92072 CB0W8K 46885950 Ki = 47.96 nM T92072 CP9G2T 46885951 Ki = 3.21 nM T92072 CU7A4P 46885952 Ki = 0.03 nM T92072 C7Y8UP 46885953 Ki = 0.19 nM T92072 C8D1QP 46885990 Ki = 0.4 nM T92072 C0TGQ9 46885991 Ki = 6.13 nM T92072 C4ELG9 46885992 Ki = 2.62 nM T92072 CH1W2C 46886345 EC50 = 4.571 nM T92072 C5EGF2 46887668 Ki = 620 nM T92072 C0S7BL 46887669 Ki = 243 nM T92072 CA41WQ 46887671 Ki = 128 nM T92072 C0TF5V 46887672 Ki = 76.8 nM T92072 CQP3K6 46887673 Ki = 42.1 nM T92072 C9PS5C 46888223 Ki = 290 nM T92072 C6NCF2 46888282 Ki = 1580 nM T92072 CR6T2J 46888283 Ki = 150 nM T92072 C2SX3E 46888356 Ki = 1170 nM T92072 C7YGA4 46888359 Ki = 960 nM T92072 CZXY41 46888782 Ki = 194 nM T92072 C0ZI2J 46888783 Ki = 203 nM T92072 C3PO0V 46888784 Ki = 159 nM T92072 CNJ6O8 46888821 Ki = 337 nM T92072 CM4KX9 46888822 Ki = 57.3 nM T92072 CS6YQ2 46888823 Ki = 12.7 nM T92072 C7F0ZH 46888824 Ki = 15.4 nM T92072 CPU7O1 46888850 Ki = 46.7 nM T92072 CR76TD 46888851 Ki = 142 nM T92072 CP3M2V 46888852 Ki = 16.4 nM T92072 CZY0H4 46888879 Ki = 32.4 nM T92072 CXEM23 46888880 Ki = 253 nM T92072 C6PEB7 46888881 Ki = 137 nM T92072 C1DOU2 46888889 Ki = 0.5 nM T92072 CY9HA1 46888890 Ki = 40 nM T92072 C27AJV 46888923 Ki = 468 nM T92072 CLA81S 46888924 Ki = 600 nM T92072 CQK1W2 46888929 Ki = 6.9 nM T92072 CJI92H 46888930 Ki = 16.4 nM T92072 CW3GP5 46888987 Ki = 172 nM T92072 CJ40AW 46888988 Ki = 119 nM T92072 C3HTX6 46888989 Ki = 107 nM T92072 CI6WP9 46888990 Ki = 40.8 nM T92072 CGE3Q5 46888991 Ki = 94.2 nM T92072 CLVB51 46889017 Ki = 34.1 nM T92072 C6LOJ5 46889018 Ki = 95.2 nM T92072 CZD9E7 46889019 Ki = 155 nM T92072 CW8UG0 46889042 Ki = 75 nM T92072 CMK23N 46889043 Ki = 140 nM T92072 CFJG37 46889044 Ki = 12.5 nM T92072 C5B2MH 46889068 Ki = 26.3 nM T92072 CP87LM 46889069 Ki = 20.4 nM T92072 CSFA02 46889070 Ki = 95.7 nM T92072 CG1YE0 46889071 Ki = 86.2 nM T92072 CP0JK9 46889095 Ki = 225 nM T92072 C45LRI 46889096 Ki = 114 nM T92072 C4P8EK 46889097 Ki = 73 nM T92072 CN51XZ 46889098 Ki = 1.8 nM T92072 CA3G2B 46889125 Ki = 17 nM T92072 CUZW61 46889126 Ki = 66.2 nM T92072 CIU27M 46889127 Ki = 20 nM T92072 CT6F8I 46889171 Ki = 208 nM T92072 C1SKA9 46889172 Ki = 94.7 nM T92072 C4HFX9 46889173 Ki = 45.2 nM T92072 CFP4E5 46889174 Ki = 215 nM T92072 CS4L1B 46889205 Ki = 258 nM T92072 C0ZJ5W 46889206 Ki = 119 nM T92072 CQSP94 46889207 Ki = 12.3 nM T92072 CE43BM 46889228 Ki = 101 nM T92072 C7PO4J 46889229 Ki = 67.4 nM T92072 CF7I9L 46889230 Ki = 191 nM T92072 CI67DB 46889231 Ki = 84.1 nM T92072 CG1AU4 46889252 Ki = 33.3 nM T92072 C83ZFB 46889253 Ki = 37.4 nM T92072 CMJ61R 46889254 Ki = 103 nM T92072 C9NHC7 46889255 Ki = 414 nM T92072 C4O0IB 46889256 Ki = 187 nM T92072 CUFE02 46893147 Ki > 1000 nM T92072 C5P0SJ 46905939 EC50 = 8300 nM T92072 CS4EX0 46905940 EC50 = 8300 nM T92072 C3JCB1 46911060 Ki = 100 nM T92072 C1LCB2 46912311 Ki = 150 nM T92072 C3H4CM 46912312 Ki = 53 nM T92072 CNU1T6 46912313 Ki = 160 nM T92072 CDTQ70 46912314 Ki = 192 nM T92072 C1BJF7 46912315 Ki = 34 nM T92072 CH79VN 47069386 Ki = 61659.5 nM T92072 CJ6EI3 47175612 Ki = 346.74 nM T92072 CAQ1Y3 49771648 IC50 = 970 nM T92072 CL4XV5 49771651 IC50 = 1600 nM T92072 CXML97 49796113 EC50 = 4500 nM T92072 CFZU73 49796118 EC50 = 17000 nM T92072 C9CH4S 49796119 EC50 = 38000 nM T92072 C29GFQ 49796975 EC50 = 36700 nM T92072 CW1G9R 49796976 EC50 > 10000 nM T92072 CW12EQ 49796978 EC50 > 10000 nM T92072 CY75IE 49796979 EC50 = 36700 nM T92072 CEFS28 49796980 EC50 > 10000 nM T92072 C79OGD 49796981 EC50 > 4200 nM T92072 CASK40 49796983 EC50 = 13300 nM T92072 CTYF79 49796984 EC50 > 10000 nM T92072 CM64ZG 49796986 EC50 = 10000 nM T92072 CQ9A0C 49796987 EC50 > 13000 nM T92072 CM34LS 49796988 EC50 = 43500 nM T92072 C2FY3G 49796989 EC50 = 19300 nM T92072 C7U3SK 49796991 EC50 = 30100 nM T92072 C5C1YE 49796992 EC50 > 8700 nM T92072 C5W9LA 49796993 EC50 > 10000 nM T92072 C3S2FN 49796996 EC50 > 10000 nM T92072 CE6HS9 49796997 EC50 = 11800 nM T92072 C9V8IS 49797004 EC50 = 13200 nM T92072 CO09NB 49797005 EC50 = 8000 nM T92072 CB16QX 49797009 EC50 > 10000 nM T92072 C8AL9C 49797010 EC50 = 11400 nM T92072 CE6C0B 49797019 EC50 = 1600 nM T92072 CG63LK 49797020 EC50 = 18000 nM T92072 CGZA72 49797026 EC50 = 34400 nM T92072 C5X0QY 49797027 EC50 > 10000 nM T92072 CHR25Y 49797032 EC50 > 10000 nM T92072 CTSR98 49797034 EC50 > 10000 nM T92072 CD7VU2 49797037 EC50 = 11800 nM T92072 C02HEX 49797747 Ki = 160 nM T92072 CC61BT 49797748 Ki = 300 nM T92072 C8HA0Y 49797749 Ki = 78 nM T92072 C6XFQ7 49797750 Ki = 130 nM T92072 CP1I3U 49797771 Ki = 150 nM T92072 CN4UQ9 49797772 Ki = 400 nM T92072 CF32QB 49797773 Ki = 410 nM T92072 CB0X1S 49797774 Ki = 110 nM T92072 C21IWV 49797793 Ki = 185 nM T92072 C4Y0JV 49797794 Ki = 71 nM T92072 C6X5LC 49797795 Ki = 390 nM T92072 CD26ZY 49797796 Ki = 30 nM T92072 CN58DG 49797797 Ki = 1600 nM T92072 CY1XE9 49797825 Ki = 790 nM T92072 CXJV63 49797826 Ki = 560 nM T92072 C4JX9B 49797827 Ki = 2600 nM T92072 CXH10P 49797828 Ki = 23 nM T92072 CF0H2A 49797852 Ki = 100 nM T92072 C7SH3X 49797853 Ki = 450 nM T92072 C7DM9C 49797854 Ki = 30 nM T92072 CB87EF 49797855 Ki = 42 nM T92072 C8FD9E 49797878 Ki = 37 nM T92072 CNRX41 49797879 Ki = 35 nM T92072 CO69IE 49797905 Ki = 6 nM T92072 C9AVX7 49797906 Ki = 9 nM T92072 CSB23K 49798137 Ki = 50 nM T92072 CJ15VM 49798138 Ki = 185 nM T92072 CEC37Y 49798139 Ki = 120 nM T92072 C7P6DN 49798140 Ki = 180 nM T92072 CZIB48 49798161 Ki = 181.97 nM T92072 CJ8CH9 49863226 Ki = 2965 nM T92072 CW1I8V 49864320 Ki = 1200 nM T92072 C3J7QB 49864672 Ki = 90 nM T92072 C84BSL 49864673 Ki = 92 nM T92072 C2GP3F 49864677 Ki = 780 nM T92072 C4OB0D 49864730 Ki = 230 nM T92072 CR14MY 49864731 Ki = 77 nM T92072 C7I2SE 49864732 Ki = 300 nM T92072 CY8B6L 49864733 Ki = 1700 nM T92072 C5YQM7 49870825 Ki = 11.4 nM T92072 CFX9W2 49870826 Ki = 47.4 nM T92072 CN5P7B 49870827 Ki = 92.7 nM T92072 CYKD61 49870828 Ki = 85.3 nM T92072 CJI59X 50751023 Ki = 10715.19 nM T92072 C4WXE2 50925499 Ki = 19 nM T92072 C0OQI7 50940921 Ki = 505 nM T92072 C1UMB4 50940926 Ki = 48.2 nM T92072 CTW9D3 50940928 Ki = 535 nM T92072 CCD60O 50940932 Ki = 367 nM T92072 CAN28T 50940939 Ki = 23.5 nM T92072 C17WCS 50940941 Ki = 678 nM T92072 CY3QD4 50940944 Ki = 255 nM T92072 CIZ5W0 50940962 Ki = 17 nM T92072 CD1U2T 50940964 Ki = 40.7 nM T92072 CZ4WU9 50940972 Ki = 83.9 nM T92072 CGYR73 50940973 Ki = 113 nM T92072 C7CH3U 50940974 Ki = 31.6 nM T92072 CJC06P 50940976 Ki = 5.28 nM T92072 CB5TZ6 50940978 Ki = 15.5 nM T92072 CMF2S3 50940979 Ki = 32.9 nM T92072 C5H8FK 50940980 Ki = 132 nM T92072 CW76LB 50940981 Ki = 39.4 nM T92072 CEZM81 50940986 Ki = 82.3 nM T92072 C8X1BV 50940988 Ki = 41.3 nM T92072 CPB75Y 50940989 Ki = 18.7 nM T92072 CL1E8H 50941003 Ki = 9.7 nM T92072 C1B7TN 50941005 Ki = 7.8 nM T92072 CLE1G9 50941006 Ki = 33.3 nM T92072 CY4W7P 50941007 Ki = 65.1 nM T92072 C15IYP 50941008 Ki = 65.1 nM T92072 C2J0GZ 51039221 Ki = 86.7 nM T92072 CPY2L4 51039223 Ki = 769 nM T92072 CUB5G9 51040798 Ki = 6900 nM T92072 CZ2NF4 51050120 Ki = 220 nM T92072 COM32L 51050226 Ki = 580 nM T92072 C3ACR2 51050227 Ki = 220 nM T92072 C8P3IT 51050841 Ki = 5400 nM T92072 C96NLK 51050843 Ki = 3730 nM T92072 C32PZT 51050844 Ki = 3890 nM T92072 CYBC20 51050845 Ki = 344 nM T92072 CO3N1B 51050939 Ki = 963 nM T92072 CGCI34 51050940 Ki = 1580 nM T92072 C35FWV 51050941 Ki = 655 nM T92072 CBX3Q5 51050942 Ki = 1010 nM T92072 CRPE85 51050944 Ki = 3510 nM T92072 CG5P0M 51051040 Ki = 991 nM T92072 C37NQZ 51051140 Ki = 1350 nM T92072 CP4Q8Y 51051143 Ki = 2950 nM T92072 CK12HU 51051145 Ki = 7470 nM T92072 CR2TW4 51051249 Ki = 1410 nM T92072 C1DB8M 51051251 Ki = 1800 nM T92072 C8Z0NV 52912216 Ki = 13 nM T92072 CYT38J 52933189 Ki > 1000 nM T92072 C8W2MH 52933190 Ki = 630 nM T92072 CMHX43 52933191 Ki = 2.2 nM T92072 C3DUB0 52933192 Ki = 36 nM T92072 C0JLH3 52933436 Ki > 1000 nM T92072 C73HZF 52933688 Ki > 1000 nM T92072 CC46SH 52933690 Ki = 59 nM T92072 CU10AR 52933691 Ki = 12 nM T92072 CYQG26 52933692 Ki = 10.5 nM T92072 C8SX6V 52933926 Ki = 0.28 nM T92072 COV1R3 52934151 Ki = 74 nM T92072 CX5K3G 52934152 Ki = 9.6 nM T92072 C71JZH 52934382 Ki = 3.6 nM T92072 CO0FQ2 52936155 Ki = 120 nM T92072 CUL5M0 52936156 Ki = 13 nM T92072 CX27DY 52940754 IC50 = 568 nM T92072 CT53UX 52941201 Ki = 377 nM T92072 CSGQ69 52941244 Ki = 170 nM T92072 C3Z5TQ 52941354 IC50 = 27 nM T92072 C36UQF 52941463 IC50 = 40 nM T92072 C9H3FM 52941478 IC50 = 435 nM T92072 C71HWB 52941597 Ki > 10000 nM T92072 CF4P2S 52941986 IC50 = 306 nM T92072 C70GZP 52942160 IC50 = 231 nM T92072 CQF4X5 52942334 Ki = 192.3 nM T92072 C3J6FO 52942359 Ki = 1370 nM T92072 CCJP23 52942475 Ki = 5999 nM T92072 CV8EW1 52942501 Ki = 1129 nM T92072 CF06HD 52942696 IC50 = 3.16 nM T92072 CNPD89 52943141 Ki = 3080 nM T92072 CW5RI6 52943163 IC50 = 1.39 nM T92072 CZ5Y2Q 52943519 Ki = 475.2 nM T92072 C2BJZ3 52943652 Ki = 15 nM T92072 CN10RU 52943791 Ki > 10000 nM T92072 C8NER0 52943888 Ki > 10000 nM T92072 C9UCH2 52944320 Ki = 3245 nM T92072 CT0Y9I 52944659 Ki = 1616 nM T92072 CEO93J 52944665 Ki = 10.2 nM T92072 C5I4BV 52944930 Ki = 101 nM T92072 CVB60F 52945006 Ki = 6050 nM T92072 C2H9AY 52945064 Ki = 7027 nM T92072 CJAY05 52945098 Ki = 159 nM T92072 C45SQC 52945195 Ki = 6.1 nM T92072 CMJ8I5 52945566 Ki = 2385 nM T92072 CNQ14E 52945627 IC50 = 294 nM T92072 CXUJ05 52945912 Ki = 252.3 nM T92072 C79TAX 52945914 Ki = 188.5 nM T92072 CHT4Z6 52946113 Ki = 68 nM T92072 CX9G3T 52946114 Ki = 183 nM T92072 CK76UG 52946159 Ki = 3253 nM T92072 CEFW97 52946211 IC50 = 3.2 nM T92072 CUA1O9 52946453 Ki = 13 nM T92072 CTMD37 52946765 Ki = 563.5 nM T92072 CE4CV0 52946784 Ki = 2445 nM T92072 CXWB47 52947034 IC50 = 233 nM T92072 C28VAP 52947301 Ki = 497 nM T92072 C7HY0V 52947452 Ki = 811 nM T92072 CV9D1Y 52947525 IC50 = 2.8 nM T92072 C4B9LU 52947745 Ki = 122.9 nM T92072 C5HLT3 52947997 Ki = 1595 nM T92072 C48RAD 52948327 Ki = 1432 nM T92072 C8Q3UH 52948332 Ki = 3920 nM T92072 C4FJ8P 52948414 Ki = 180.2 nM T92072 C6JN5H 52948418 Ki = 71.8 nM T92072 C4KA6Y 52948671 Ki = 3623 nM T92072 COW0J3 52948763 Ki = 10443 nM T92072 C3B9OG 52948788 IC50 = 9 nM T92072 C7TI2R 52948915 Ki = 1153 nM T92072 C28MQF 52948949 Ki = 68 nM T92072 CQ91YN 52948995 IC50 = 13 nM T92072 C6ZXI9 52949641 Ki = 267.4 nM T92072 C2MAQ9 52949644 Ki = 28.3 nM T92072 C67NOY 52949655 Ki = 43.6 nM T92072 CE8F3G 52949755 Ki = 3914 nM T92072 CE3XQ7 52949772 Ki = 8603 nM T92072 CL6K9M 52949999 Ki = 602 nM T92072 C74BRO 52950000 Ki = 1085 nM T92072 CHM1G6 52950027 Ki = 436 nM T92072 C0L8VT 52950028 Ki = 1720 nM T92072 CQAP62 52950040 Ki = 8.6 nM T92072 C3JEO8 52950206 Ki = 1334 nM T92072 C7DWU2 53131655 Ki = 588.84 nM T92072 CRB59S 53242165 Ki = 690 nM T92072 CI35WL 53248698 Ki = 100 nM T92072 CDS80Q 53248700 Ki = 19 nM T92072 CD07TO 53258079 Ki = 140 nM T92072 C0VX3M 53258080 Ki = 300 nM T92072 CKV8G6 53258081 Ki = 100 nM T92072 CE3C7M 53258185 Ki = 455 nM T92072 CJZ98W 53318744 Ki = 27 nM T92072 CH7O8A 53324032 Ki = 130 nM T92072 CN51SY 53348048 Ki > 10000 nM T92072 C7NOK1 53353232 Ki = 194.98 nM T92072 CIVP28 53354521 Ki = 56.23 nM T92072 CIAO19 53354627 Ki = 10000 nM T92072 CH6X9F 53354632 Ki = 43.65 nM T92072 C45VUI 53354728 Ki = 10000 nM T92072 CL3P8I 53394567 Ki = 2220 nM T92072 CPY9J6 53587504 Ki = 29512.09 nM T92072 CUO97T 54577823 Ki = 7130 nM T92072 CZQ2H9 54580150 Ki = 10 nM T92072 C9LU8J 54580623 Ki > 100000 nM T92072 CT1CO5 54580654 Ki = 1100 nM T92072 C84FJX 54581142 Ki = 6 nM T92072 CSX07T 54581143 Ki = 31 nM T92072 CX3Y6L 54581663 Ki = 1000 nM T92072 C85ZXD 54582166 Ki = 61 nM T92072 C2C8MB 54582167 Ki = 67 nM T92072 CHDV60 54583133 Ki = 220 nM T92072 CHXE36 54583615 Ki = 4840 nM T92072 C08HKQ 54583616 Ki = 1300 nM T92072 CSF9W8 54583714 Ki = 1700 nM T92072 CS6O9E 54584124 Ki = 2 nM T92072 C7CWY9 54584125 Ki = 78 nM T92072 CP04UN 54584599 Ki = 1270 nM T92072 C2BOV8 54584981 IC50 = 2800 nM T92072 C3N7RC 54585057 Ki = 7 nM T92072 CO7IC0 54585058 Ki = 5 nM T92072 CKCD81 54585511 Ki = 22100 nM T92072 C6UMY3 54585937 IC50 = 1900 nM T92072 C02CVB 54586036 Ki = 120 nM T92072 C6IV3L 54587015 Ki = 220 nM T92072 CSL08D 54587662 Ki = 932 nM T92072 C83VFS 54754508 Ki = 6490 nM T92072 C40IVD 54768079 Ki > 10000 nM T92072 C1UW4E 54768080 Ki > 10000 nM T92072 C4JA9T 54768112 Ki > 10000 nM T92072 C2JPC3 54768115 Ki > 10000 nM T92072 CL5SE3 54768601 Ki > 10000 nM T92072 C6SYD1 54768602 Ki > 10000 nM T92072 CX9A4R 54768635 Ki = 10300 nM T92072 C3HNS6 54768636 Ki > 10000 nM T92072 CB7T1O 56627882 Ki = 0.966 nM T92072 C6WSF9 56657920 Ki > 100000 nM T92072 CD7C2P 56661442 Ki = 221 nM T92072 C2FI4U 56661443 Ki = 831 nM T92072 CZ6I4O 56662964 Ki = 970 nM T92072 CVLM74 56664888 Ki > 100000 nM T92072 CBQS24 56668308 Ki = 395 nM T92072 CYNJ53 56668410 Ki > 100000 nM T92072 CWM34N 56668411 Ki = 12900 nM T92072 CSJ34D 56668412 Ki > 30000 nM T92072 C98FPH 56671922 Ki > 100000 nM T92072 CD6C0P 56675199 Ki > 100000 nM T92072 CH8YR5 56675200 Ki = 192 nM T92072 CUJ34X 56675201 Ki = 232 nM T92072 CK3AZ9 56675297 Ki = 5550 nM T92072 C58FTQ 56675298 Ki > 10000 nM T92072 C7TNW9 56675299 Ki > 30000 nM T92072 CDN69Q 56678498 Ki > 10000 nM T92072 C13UZX 56678638 Ki > 30000 nM T92072 CM04LK 56678639 Ki = 4420 nM T92072 CVP0A9 56681843 Ki > 10000 nM T92072 C02DIY 56838950 Ki = 541 nM T92072 CYS17U 56844240 Ki = 85.11 nM T92072 COY13J 56924646 Ki = 733 nM T92072 C86NML 56935713 Ki = 36 nM T92072 CF60KW 56943766 Ki = 1700 nM T92072 C8TZ4I 56944263 Ki = 5000 nM T92072 CB7I4R 56945639 Ki = 740 nM T92072 C9XFM7 56945648 Ki = 1080 nM T92072 CCK34B 56945649 Ki = 1230 nM T92072 C3WC9H 56945650 Ki = 1670 nM T92072 C5DT0Z 56945768 Ki = 1610 nM T92072 CU4C5D 56945769 Ki = 1900 nM T92072 CR1YL9 56945770 Ki = 1180 nM T92072 CPA2Z6 56945771 Ki = 1110 nM T92072 CY4D9S 56945868 Ki = 290 nM T92072 C9J2PL 56945870 Ki = 500 nM T92072 CKZE52 56945888 Ki = 990 nM T92072 C9VLJ0 56945889 Ki = 640 nM T92072 CRF5J8 56945890 Ki = 550 nM T92072 CX3W2C 56945891 Ki = 1060 nM T92072 CD4ZW9 56945994 Ki = 2160 nM T92072 CI0Q2T 56945995 Ki = 1000 nM T92072 CR5AJ1 56945996 Ki = 350 nM T92072 CH1JR4 56950235 Ki = 800 nM T92072 CXB8Z6 56951623 Ki = 140 nM T92072 C9F7YE 56954252 Ki = 0.5 nM T92072 CTXB04 56954253 Ki = 1.8 nM T92072 C70KFB 56954254 Ki = 29.3 nM T92072 CL56UR 56954333 Ki = 223 nM T92072 CLTD39 56954334 Ki = 5.2 nM T92072 CIJN02 56954335 Ki = 6 nM T92072 CH5A4T 56954336 Ki = 2.5 nM T92072 CH3GM5 56964225 Ki = 31 nM T92072 C9T1XQ 56964459 Ki = 1357 nM T92072 CY1IG3 56964460 Ki > 10000 nM T92072 CZ42XV 56964461 Ki > 10000 nM T92072 CC50SG 56964576 Ki > 10000 nM T92072 CHR8L5 57325914 Ki > 10000 nM T92072 C7SRT3 57325915 Ki > 10000 nM T92072 CREU79 57328471 Ki > 100000 nM T92072 C8JY3E 57384287 IC50 = 2324 nM T92072 CYSA75 57384288 IC50 = 3990 nM T92072 CDN54M 57384289 IC50 = 2136 nM T92072 CA63RT 57384543 IC50 = 2208 nM T92072 CW63IC 57384544 IC50 = 5251 nM T92072 CCPY02 57385043 IC50 = 3914 nM T92072 CKO3L1 57387337 IC50 = 0.36 nM T92072 C8X7MO 57387594 IC50 = 10 nM T92072 C6XKL9 57387596 IC50 = 122 nM T92072 C7XW0T 57387822 IC50 = 413267 nM T92072 CT1R6Q 57387824 IC50 = 326 nM T92072 C01AHY 57387825 IC50 = 2082 nM T92072 CNL3P2 57388054 IC50 = 1007 nM T92072 CK7R6O 57388055 IC50 = 1184 nM T92072 CMBN74 57388056 IC50 = 428 nM T92072 CD52CA 57391118 IC50 = 440 nM T92072 C1BAX6 57391653 Ki = 18 nM T92072 C45GCN 57391694 Ki = 33 nM T92072 C03HUE 57391695 Ki = 12 nM T92072 CJF61Z 57391696 Ki > 1000 nM T92072 CC3X7G 57393433 Ki = 524 nM T92072 C1B3QM 57393434 Ki > 1000 nM T92072 C8ZX4L 57393435 Ki > 1000 nM T92072 CVO2P8 57395120 Ki = 743 nM T92072 C9VWH7 57395161 Ki = 355 nM T92072 CJM7E8 57395162 Ki = 85 nM T92072 CEQR05 57395163 Ki = 129 nM T92072 CDP13M 57395164 Ki = 923 nM T92072 CSTG21 57396888 Ki = 4.3 nM T92072 CWX64M 57396935 Ki = 10 nM T92072 CC52TB 57396936 Ki = 22 nM T92072 C1WT0H 57396937 Ki > 1000 nM T92072 CD6JT5 57398641 Ki = 35 nM T92072 CHC8U6 57398676 Ki = 7.1 nM T92072 C1J3DG 57400352 Ki = 14 nM T92072 CNRY34 57400353 Ki = 240 nM T92072 CIX58U 57402117 Ki = 100 nM T92072 CLCX61 57402118 Ki = 178 nM T92072 CBMP08 57402160 Ki = 210 nM T92072 C58APE 57402161 Ki = 30 nM T92072 CKB51R 57402162 Ki = 753 nM T92072 CQK46U 57402163 Ki > 1000 nM T92072 CYHD10 57403904 Ki = 61 nM T92072 CD2NO5 57403905 Ki = 4.9 nM T92072 C05DRY 57429649 Ki = 177 nM T92072 C4IQ0H 57523214 Ki = 1520 nM T92072 C7F4QX 57524978 Ki = 383 nM T92072 C4GZY7 58739995 Ki = 323 nM T92072 C1HU4O 59011969 Ki = 7240 nM T92072 CK7T6D 59179887 IC50 > 1000 nM T92072 CY0J5M 59276682 Ki = 740 nM T92072 CB31TY 59276704 Ki = 17820 nM T92072 C92ZHB 59276711 Ki = 330 nM T92072 C1EWD7 59277997 Ki = 493 nM T92072 CF60BK 59277999 Ki = 1159 nM T92072 C5G2RH 60154738 Ki = 614 nM T92072 C4U7BI 60154739 Ki = 396 nM T92072 CU3R2Q 60154740 Ki = 635 nM T92072 CJ57XU 60154742 Ki = 1299 nM T92072 CUK15D 60154835 Ki = 1123 nM T92072 CK7VH4 60154837 Ki = 3408 nM T92072 C3PO4T 60155712 Ki > 5000 nM T92072 CJB03P 60155713 Ki > 5000 nM T92072 C6W8XE 60155714 Ki = 2794 nM T92072 CN03ZC 60155715 Ki = 3357 nM T92072 CEZ4V5 60155716 Ki = 802 nM T92072 C1ZXO7 60155796 Ki = 703 nM T92072 CZRU45 60155797 Ki = 1049 nM T92072 C8GZ3V 60155798 Ki = 724 nM T92072 CXLO10 60155799 Ki = 1478 nM T92072 CYB1L4 60155893 Ki = 1156 nM T92072 C0B5OZ 60155894 Ki = 166 nM T92072 CB9A6F 60155895 Ki = 371 nM T92072 C2VPM8 60155896 Ki = 1329 nM T92072 CW7R1L 60155897 Ki = 1188 nM T92072 CP3H2Z 60156002 Ki = 348 nM T92072 C8KU5V 60156003 Ki = 1500 nM T92072 C2LN4J 60156004 Ki = 1324 nM T92072 C8SZE0 60156005 Ki = 744 nM T92072 CGL84Y 60156006 Ki = 761 nM T92072 CFBG07 60156104 Ki = 805 nM T92072 CKVJ21 60156105 Ki = 525 nM T92072 C7L1BF 60156106 Ki = 182 nM T92072 C38NUA 60156107 Ki = 112 nM T92072 C87SMR 60156108 Ki = 408 nM T92072 CEI9G2 60194835 EC50 > 10000 nM T92072 CAD2Y0 60194917 EC50 = 530 nM T92072 CH3E7Z 60194919 EC50 = 6100 nM T92072 CD9O1E 60194921 EC50 = 4400 nM T92072 CXBY52 60195011 EC50 = 550 nM T92072 C16CSN 60195998 EC50 = 21 nM T92072 CQAR83 60196082 EC50 = 100 nM T92072 CF2ZS0 60196083 EC50 = 5400 nM T92072 C7UCR6 60196155 EC50 = 1500 nM T92072 CIU75L 60196156 EC50 > 10000 nM T92072 CJE1H0 60196158 EC50 = 120 nM T92072 CF1PG5 60741010 Ki = 12302.69 nM T92072 CLM18K 66678431 Ki = 24 nM T92072 C20XJH 66892244 Ki = 711 nM T92072 CWN0X9 66892382 Ki = 340 nM T92072 CV6PW1 66892867 Ki = 346 nM T92072 C9GDP5 66894241 Ki = 108 nM T92072 C5SVP6 67192387 Ki > 1000 nM T92072 C0L8HB 67192741 Ki = 2.3 nM T92072 CO94DL 67193593 Ki = 27 nM T92072 CT32UQ 67195703 Ki = 5.5 nM T92072 CTE5F4 67195808 Ki = 4500 nM T92072 C1XZV9 67364057 Ki = 398.11 nM T92072 C41MUQ 67364090 Ki = 169.82 nM T92072 CXQL59 67364157 Ki = 117.49 nM T92072 CS0D4B 67364791 Ki = 109.65 nM T92072 CW37UH 67548131 IC50 = 537 nM T92072 C56UIN 67548175 IC50 = 399 nM T92072 C6VKP4 67548337 IC50 = 28 nM T92072 CGXY26 67548392 IC50 = 61 nM T92072 C5U3WL 67548498 IC50 = 184 nM T92072 C6LA7R 67548508 IC50 = 2 nM T92072 CC4Y6V 67548720 IC50 = 5 nM T92072 C8B1JS 67548983 IC50 = 634 nM T92072 CPQ2I7 67549056 IC50 > 1000 nM T92072 C71HZU 67549086 IC50 = 31 nM T92072 C74YXW 67549097 IC50 = 324 nM T92072 CD09WI 67549451 IC50 = 59 nM T92072 C5M0NT 67549626 IC50 > 1000 nM T92072 C8Z7RX 67549879 IC50 > 1000 nM T92072 C18CNK 68405754 IC50 = 71 nM T92072 CNYS04 68405874 IC50 = 81 nM T92072 CWEQ54 68405927 IC50 > 1000 nM T92072 C2OM6I 69029783 Ki > 800 nM T92072 CRL75S 69031481 Ki = 670 nM T92072 C0P1OR 69427076 Ki = 8.4 nM T92072 C32SHY 69612603 IC50 = 2.9 nM T92072 CXUB67 69846372 Ki = 2270 nM T92072 C76KTS 69846756 Ki = 5720 nM T92072 CY26GL 69937963 Ki > 1000 nM T92072 CCDH27 69961639 Ki = 52 nM T92072 C5FG6U 70655621 Ki = 85 nM T92072 CQ90VH 70655647 Ki = 23 nM T92072 CXM72L 70655818 Ki = 50 nM T92072 CUN7P5 70655981 Ki = 5.9 nM T92072 C1EJX7 70656885 Ki > 1000 nM T92072 CAH95Y 70660748 Ki > 1000 nM T92072 CAN39T 70660767 Ki = 370 nM T92072 C1Q3ST 70676457 Ki = 780 nM T92072 CJ7Y1S 70676459 Ki = 68.1 nM T92072 COVC42 70676460 Ki = 150 nM T92072 C9OLG0 70676461 Ki = 76 nM T92072 CCO40K 70676610 Ki = 150 nM T92072 C21ANJ 70676611 Ki = 270 nM T92072 CN38XM 70676612 Ki = 120 nM T92072 CYTH16 70676613 Ki = 490 nM T92072 C0VI8J 70676614 Ki = 170 nM T92072 C5ETD9 70676615 Ki = 3000 nM T92072 CL04EV 70677099 Ki = 56.1 nM T92072 CZA8H7 70677100 Ki = 488 nM T92072 C46HBT 70681087 Ki = 230 nM T92072 CIT56B 70681088 Ki = 78.8 nM T92072 C5W7QI 70681089 Ki = 4790 nM T92072 CE3N0Y 70681091 Ki = 1910 nM T92072 CS0I7Z 70682890 Ki = 2.7 nM T92072 C7LZO2 70683991 Ki = 2511.89 nM T92072 C0XG9F 70685288 Ki = 140 nM T92072 CK75QB 70685289 Ki = 72.7 nM T92072 CTQ61B 70685290 Ki = 86.8 nM T92072 CWE50T 70685291 Ki = 3580 nM T92072 CB4VD0 70687115 Ki = 2730 nM T92072 CM03SU 70687435 Ki = 51.6 nM T92072 CL63IQ 70687436 Ki = 68.4 nM T92072 CWC6O5 70687437 Ki = 1260 nM T92072 C1KJD5 70689262 Ki = 340 nM T92072 C7X1UJ 70689496 Ki = 350 nM T92072 C4U2AE 70689497 Ki = 760 nM T92072 CA4E1B 70690267 Ki = 6309.57 nM T92072 C58QIA 70691614 Ki = 200 nM T92072 CDP9H6 70693700 Ki = 930 nM T92072 C1KHZ2 70694510 Ki = 545 nM T92072 CGW8U4 70695809 Ki = 210 nM T92072 CL3E6M 70695810 Ki = 82.6 nM T92072 C26LVT 70695811 Ki = 72.2 nM T92072 CVU08A 70695812 EC50 = 40.7 nM T92072 C7USK0 70696572 Ki = 404 nM T92072 CBN9A8 70697521 Ki = 1.5 nM T92072 CGXQ60 71041800 IC50 = 2340 nM T92072 C3J4SN 71041846 IC50 > 10000 nM T92072 C75JTG 71361867 Ki = 42800 nM T92072 CAR92Q 71364275 Ki = 4640 nM T92072 C31FGM 71412032 Ki = 14 nM T92072 C4O3XF 71449066 Ki = 2600 nM T92072 CBZM95 71449068 Ki = 190 nM T92072 CXZ40U 71450227 Ki = 711 nM T92072 C38UKP 71450240 Ki = 6560 nM T92072 CXM83Y 71450241 Ki = 1930 nM T92072 C9G0FP 71450242 Ki = 223 nM T92072 CC73UY 71450243 Ki = 484 nM T92072 CTYM41 71450845 Ki = 640 nM T92072 C37NIO 71450846 Ki = 2600 nM T92072 CW75JC 71450849 Ki = 34.1 nM T92072 CPQ4Y9 71451659 Ki = 730 nM T92072 C4LVT1 71452054 Ki = 2150 nM T92072 CC2Q9H 71452055 Ki = 1020 nM T92072 CQ4CA3 71452056 Ki = 338 nM T92072 CWOB13 71452072 Ki = 248 nM T92072 CX52PV 71452672 Ki = 540 nM T92072 CXF65C 71452801 Ki = 8 nM T92072 C0NC4G 71453140 Ki > 10000 nM T92072 C9QD3W 71453871 Ki = 639 nM T92072 CKW2G6 71453872 Ki = 15000 nM T92072 C0VK4E 71453873 Ki = 328 nM T92072 CR8A0V 71453874 Ki = 527 nM T92072 CV0NW6 71453875 Ki = 1230 nM T92072 C5S3FU 71453891 Ki = 212 nM T92072 C0M9CP 71453892 Ki = 604 nM T92072 CY1B4N 71453893 Ki = 982 nM T92072 C76PJS 71453894 Ki = 166 nM T92072 CO02WB 71454439 Ki = 710 nM T92072 C56VEI 71455599 Ki = 483 nM T92072 C79IVN 71455600 Ki = 2400 nM T92072 CM2ZF9 71455601 Ki = 646 nM T92072 CEO64T 71455602 Ki = 4760 nM T92072 CPN0B7 71455603 Ki = 538 nM T92072 CUE71P 71455604 Ki = 442 nM T92072 CC1RD4 71455619 Ki = 1580 nM T92072 C2ITP7 71455620 Ki = 133 nM T92072 CQ8U5S 71455621 Ki = 165 nM T92072 CB2E9C 71455622 Ki = 481 nM T92072 CTH1W7 71455623 Ki = 605 nM T92072 C1QLP9 71455624 Ki = 169 nM T92072 CVJZ12 71456194 Ki = 1600 nM T92072 CJBC05 71456195 Ki = 770 nM T92072 C4J0QI 71456197 EC50 = 1 nM T92072 C5BHA3 71457388 Ki = 1040 nM T92072 CYTZ37 71457389 Ki = 2750 nM T92072 C3H2QF 71457390 Ki = 945 nM T92072 CPBO67 71457391 Ki = 322 nM T92072 C12PEI 71457403 Ki = 649 nM T92072 C19MUP 71457404 Ki = 333 nM T92072 CS6Z4N 71457405 Ki = 131 nM T92072 C5RD0O 71457406 Ki = 265 nM T92072 C6MF5O 71457407 Ki = 80.1 nM T92072 CG1P7Y 71457987 EC50 = 1.1 nM T92072 CJA6M2 71457990 Ki = 610 nM T92072 C0DPK5 71457992 Ki = 1600 nM T92072 C6QJ9D 71458047 Ki = 1470 nM T92072 CJO41A 71458816 Ki = 37.3 nM T92072 CU0YQ6 71459244 Ki = 169 nM T92072 CV3L0D 71459245 Ki = 2420 nM T92072 CDW92B 71459246 Ki = 1060 nM T92072 C5WX8S 71459247 Ki = 566 nM T92072 CN79LY 71459248 Ki = 3310 nM T92072 C82QUK 71459249 Ki = 750 nM T92072 CC9I6G 71459250 Ki = 2720 nM T92072 CQ7BP5 71459268 Ki = 1250 nM T92072 CG8MI3 71459899 Ki = 450 nM T92072 C8AY0D 71460344 Ki > 10000 nM T92072 CY0LV4 71460666 Ki = 210 nM T92072 CJ1R3V 71460667 Ki = 1080 nM T92072 CB9A8S 71461026 Ki = 525 nM T92072 C60OEP 71461027 Ki = 3330 nM T92072 CUDN57 71461028 Ki = 823 nM T92072 CJ9K0H 71461029 Ki = 17500 nM T92072 CDX9O4 71461045 Ki > 30000 nM T92072 COU59X 71461116 Ki = 104 nM T92072 CA1TQ7 71461609 Ki = 4100 nM T92072 CQ7V9L 71461900 Ki = 8100 nM T92072 CA0EJ2 71462751 Ki = 15200 nM T92072 CK7OB3 71462752 Ki = 375 nM T92072 CP07FL 71462753 Ki = 219 nM T92072 CK97MP 71462754 Ki = 1450 nM T92072 CV1QN8 71462755 Ki = 733 nM T92072 COU6E4 71462772 Ki = 7750 nM T92072 CGC23V 71462773 Ki = 129 nM T92072 C1HAS6 71462774 Ki = 208 nM T92072 CHT04N 71462775 Ki = 802 nM T92072 CGT9W5 71508481 Ki = 35 nM T92072 CNKZ09 71528098 Ki > 100000 nM T92072 CT29GM 71570217 Ki = 22.6 nM T92072 CI39JB 71601630 Ki = 70 nM T92072 C9J4OB 71601631 Ki = 75 nM T92072 CRQP84 71601632 Ki = 150 nM T92072 CE89VB 71601788 Ki = 510 nM T92072 CN2BP6 71602912 Ki = 520 nM T92072 C76WQP 71602913 Ki < 16 nM T92072 C3J1QE 71602914 Ki = 2954 nM T92072 CF4XL2 71602915 Ki = 310 nM T92072 CXD5L1 71602961 Ki = 28.6 nM T92072 CT4FI9 71603017 Ki = 237 nM T92072 C8UJ5P 71603087 Ki < 16 nM T92072 CER07O 71603088 Ki = 3713 nM T92072 C0TOS6 71603089 Ki = 812 nM T92072 C09TYA 71603090 Ki > 1000 nM T92072 CM87NU 71623050 Ki = 87 nM T92072 CNZ17D 71657835 EC50 = 42.66 nM T92072 C0YW1C 71680730 Ki > 10000 nM T92072 CK2Y6A 71680733 Ki = 2500 nM T92072 CH5KU9 71680734 Ki = 214 nM T92072 C6OXR9 71680735 Ki > 10000 nM T92072 CCM92I 71680890 Ki = 822 nM T92072 CS51FY 71680891 Ki = 500 nM T92072 CX4BZ6 71680892 Ki = 562 nM T92072 C6HZ4O 71680894 Ki > 1000 nM T92072 CN0EZ6 71680895 Ki > 1000 nM T92072 C30NCG 71681049 Ki = 4370 nM T92072 CVY85K 71681051 Ki = 1000 nM T92072 CLBD58 71681054 Ki = 785 nM T92072 C2Y3KO 71681203 Ki = 364 nM T92072 C21UWV 71683091 Ki = 1050 nM T92072 COWX82 71683092 Ki = 1370 nM T92072 C3RD0E 71713167 Ki = 14700 nM T92072 CPO02N 71716569 EC50 = 0.81 nM T92072 CG65UK 71717167 EC50 = 10 nM T92072 C1X5OE 71878818 Ki = 1949.84 nM T92072 C2CRW9 71878833 Ki = 56234.13 nM T92072 CS87DW 72164230 Ki = 0.00059 nM T92072 C8GZ5E 72164231 Ki = 101.8 nM T92072 COR6T8 72164232 Ki = 16.7 nM T92072 CTWX78 72164233 Ki = 889.2 nM T92072 CAR8I1 72164234 Ki = 0.00063 nM T92072 CXZM13 72164235 Ki = 19.82 nM T92072 CL57OG 72164236 Ki = 2.32 nM T92072 CO1R8B 72164352 Ki = 24630 nM T92072 C3H2GK 72164353 Ki = 412.7 nM T92072 C4REK7 72164354 Ki = 0.00074 nM T92072 CHQ6M0 72164355 Ki = 606.7 nM T92072 CYN8X6 72164356 Ki = 0.1 nM T92072 CLFV53 72164357 Ki = 0.25 nM T92072 C9F1AX 72164358 Ki = 186 nM T92072 C5EMX3 72197342 Ki = 688 nM T92072 C4E0QC 72197343 Ki > 10000 nM T92072 C76ASV 72197513 Ki = 3630 nM T92072 CZW4Y0 72197514 Ki = 801 nM T92072 CUL8V0 72197515 Ki > 100000 nM T92072 CXF4U1 72197516 Ki > 30000 nM T92072 C3QYT8 72197517 Ki = 7240 nM T92072 C4W8LQ 72197698 Ki > 10000 nM T92072 CY8GU4 72197699 Ki > 10000 nM T92072 C6BUC3 72197700 Ki > 10000 nM T92072 C48QTY 72197701 Ki = 406 nM T92072 C4D8WO 72197702 Ki = 177 nM T92072 CAY6J2 72197703 Ki = 276 nM T92072 C6RDT4 72197880 Ki = 0.58 nM T92072 C7XN0S 72197881 Ki = 12000 nM T92072 C5J9QH 72197882 Ki > 10000 nM T92072 CB05ET 72197883 Ki = 536 nM T92072 C52QMK 72197884 Ki > 10000 nM T92072 CWH6T3 72548703 IC50 = 0.61 nM T92072 C1E4ZD 72696146 Ki = 1700 nM T92072 CWG0U4 72697647 Ki = 3610 nM T92072 CH90JS 72697648 Ki = 9490 nM T92072 CPB7K4 72697649 Ki > 10000 nM T92072 C1D7VQ 72697650 Ki = 9650 nM T92072 CA5BI1 72697652 Ki = 249 nM T92072 C50SYX 72697785 Ki = 605 nM T92072 CXPB58 72697786 Ki = 1330 nM T92072 CJ5W1R 72697787 Ki = 10200 nM T92072 CY1I8G 72697789 Ki = 410 nM T92072 CXDT98 72697790 Ki = 11600 nM T92072 CS7VK8 72697791 Ki = 8260 nM T92072 CX69MI 72697928 Ki = 4400 nM T92072 CEWO96 72697930 Ki = 1410 nM T92072 CNP9S3 72697931 Ki = 866 nM T92072 C3NR4V 72697932 Ki = 2360 nM T92072 CQ4IE7 72697933 Ki = 1150 nM T92072 CY94KO 72697934 Ki = 1870 nM T92072 CVB0Y9 72698080 Ki = 6650 nM T92072 CZG6V9 72698083 Ki = 3920 nM T92072 CST61L 72698226 Ki = 1040 nM T92072 CJA8Q5 72713752 IC50 = 21000 nM T92072 CW83DK 73213196 Ki > 10000 nM T92072 CRO2K8 73345315 Ki = 200 nM T92072 CRW73S 73345316 Ki = 2200 nM T92072 C50TLE 73346045 IC50 = 26.92 nM T92072 C5AB9Z 73346835 Ki = 340 nM T92072 CF1JN5 73347573 Ki > 10000 nM T92072 CM5B9S 73347862 Ki = 161.5 nM T92072 CTJ0U3 73348946 Ki = 10400 nM T92072 C9ZX2M 73349104 IC50 = 128.82 nM T92072 C31QUT 73349105 IC50 = 74.13 nM T92072 C2PTH6 73349106 Ki = 9549.93 nM T92072 CK78DU 73349125 IC50 = 269.15 nM T92072 CI65VU 73349920 Ki = 1300 nM T92072 C4C0GK 73349930 Ki = 270 nM T92072 CY5K9T 73350674 Ki > 10000 nM T92072 C56YIX 73350675 EC50 = 234.42 nM T92072 C3XOK2 73350676 EC50 = 263.03 nM T92072 CHLF98 73350966 Ki > 10000 nM T92072 CE2YB8 73350967 IC50 = 291.4 nM T92072 CQSX70 73350968 Ki > 10000 nM T92072 CX82US 73352174 IC50 = 1122.02 nM T92072 C5YXO4 73352175 Ki > 10000 nM T92072 CIH36P 73352882 Ki = 81 nM T92072 C35XEH 73352883 Ki = 1200 nM T92072 C2M8PJ 73353634 Ki = 6456.54 nM T92072 CV1Q5U 73355133 IC50 = 5.248 nM T92072 CW18JX 73355444 Ki > 10000 nM T92072 C4HX2J 73355960 Ki = 48 nM T92072 CXT6Y5 75413912 Ki = 3162.28 nM T92072 CMS65T 76309882 Ki = 3000 nM T92072 CB84HP 76309883 Ki = 756 nM T92072 C02EBL 76309925 Ki > 100000 nM T92072 CX1H6Y 76310493 Ki = 9000 nM T92072 C9DL1B 76310832 Ki = 1.2 nM T92072 CCX8V6 76311194 EC50 = 251.19 nM T92072 CQLE57 76311197 EC50 = 794.33 nM T92072 CSV43U 76313599 Ki = 652 nM T92072 CP2TA1 76313600 Ki = 438 nM T92072 CQ5Z4P 76313639 Ki > 100000 nM T92072 CY8D4J 76313640 Ki > 100000 nM T92072 CB0WN9 76313641 Ki > 100000 nM T92072 C1C3LK 76314155 Ki = 2700 nM T92072 C25LDC 76314450 Ki = 1.82 nM T92072 CEO9I0 76314563 Ki = 2170 nM T92072 CZX45G 76314797 EC50 = 398.11 nM T92072 C21BCT 76317721 Ki > 100000 nM T92072 C2K6XR 76317722 Ki = 13800 nM T92072 CY3V7H 76317723 Ki > 100000 nM T92072 CXQY23 76317724 Ki = 16300 nM T92072 CCY8V2 76318040 Ki = 1.33 nM T92072 CL4JH8 76318403 EC50 = 63.1 nM T92072 C9O4CQ 76320863 Ki > 100000 nM T92072 CKLB89 76320909 Ki = 0.7 nM T92072 CL46PW 76321429 Ki = 3400 nM T92072 CWO42D 76321430 Ki = 11100 nM T92072 CFN3M9 76321431 Ki = 31900 nM T92072 CY5TN2 76321753 Ki = 1.59 nM T92072 C5R6OT 76322076 EC50 = 398.11 nM T92072 CK5Z6L 76324475 Ki = 496 nM T92072 CHWO53 76324476 Ki = 62 nM T92072 C3CE4B 76324522 Ki > 30000 nM T92072 C6AV9Z 76325026 Ki = 7900 nM T92072 C1JV7S 76325027 Ki = 6500 nM T92072 CQ51JN 76325369 Ki = 2.58 nM T92072 C2DPT3 76325370 Ki > 10 nM T92072 CP4CY1 76325371 Ki = 0.89 nM T92072 C5J4ML 76325372 Ki > 30 nM T92072 COD78V 76325693 EC50 > 10000 nM T92072 C3FE0S 76325694 EC50 = 63.1 nM T92072 CC67KO 76328082 Ki > 100000 nM T92072 CA0MJ2 76328083 Ki > 100000 nM T92072 C72UFI 76328084 Ki = 16500 nM T92072 CNM0E1 76328596 Ki > 100000 nM T92072 CXTN91 76328597 Ki > 100000 nM T92072 C3TH4J 76328598 Ki = 3800 nM T92072 CQI9X5 76328599 Ki > 60000 nM T92072 C0AE9L 76328600 Ki > 100000 nM T92072 C5B0UO 76328910 Ki = 1.85 nM T92072 C5VEJ9 76328911 Ki > 30 nM T92072 C8O5KF 76329263 EC50 = 316.23 nM T92072 C9O0UH 76329264 EC50 = 501.19 nM T92072 CF82DA 76329265 EC50 = 39.81 nM T92072 CPVN52 76329266 EC50 = 6309.57 nM T92072 C0E9DN 76330242 Ki = 7800 nM T92072 CG30CO 76331702 Ki = 19 nM T92072 C6QY2P 76331703 Ki = 922 nM T92072 CFNG34 76331754 Ki > 30000 nM T92072 CMR14L 76331755 Ki > 100000 nM T92072 CQT81A 76332277 Ki = 4300 nM T92072 CH64XC 76332278 Ki = 19600 nM T92072 CQWD47 76332279 Ki > 100000 nM T92072 CJKD34 76332280 Ki = 10800 nM T92072 C1GZ8R 76332281 Ki > 60000 nM T92072 CVT1E3 76332599 Ki > 30 nM T92072 CVS3F8 76332600 Ki > 30 nM T92072 CIF6V7 76332686 Ki = 1580 nM T92072 CYK39X 76332918 EC50 > 10000 nM T92072 C4S8NF 76332919 EC50 = 3981.07 nM T92072 CF68KC 76335303 Ki = 60 nM T92072 CL83MV 76335304 Ki = 583 nM T92072 C7KY5A 76335305 Ki = 69 nM T92072 CC5IO4 76335344 Ki = 25000 nM T92072 C7FE5D 76335345 Ki > 100000 nM T92072 CIT36F 76335346 Ki > 100000 nM T92072 CV05FX 76335917 Ki = 12000 nM T92072 CLN8S6 76335918 Ki > 100000 nM T92072 CM0D3G 76335919 Ki = 4100 nM T92072 CO86UR 76335920 Ki = 11000 nM T92072 CESR09 76335921 Ki = 16500 nM T92072 CR85PG 76335922 Ki > 100000 nM T92072 C3HE2N 76335923 Ki = 1900 nM T92072 C5DSC0 76335924 Ki > 100000 nM T92072 C5VM4Q 76336198 Ki > 30 nM T92072 CH9WJ4 76336525 EC50 = 2511.89 nM T92072 CNL62P 76336526 EC50 = 316.23 nM T92072 C5ZRE9 76336527 EC50 = 316.23 nM T92072 CIF8S6 85532110 Ki = 213 nM T92072 CI4M9P 85706712 Ki = 6280 nM T92072 CQS7X2 88448936 Ki = 5.6 nM T92072 C0M7NI 90268057 Ki = 1448 nM T92072 CY5P6I 90268061 Ki = 1095 nM T92072 C9R6LO 90644464 IC50 = 8000 nM T92072 C8TK5D 90644465 IC50 = 8000 nM T92072 CBT08V 90644466 IC50 = 8000 nM T92072 C7YTQ8 90644469 IC50 = 8000 nM T92072 CB51WQ 90654601 Ki = 9.7 nM T92072 CI2F0T 90654602 Ki = 4.8 nM T92072 CR8BK4 90654603 EC50 = 3.9 nM T92072 CF9N7J 90654604 Ki = 8.9 nM T92072 C5GI9U 90654606 Ki = 185 nM T92072 CZ6BY3 90654607 EC50 = 4.9 nM T92072 C0XE3Q 90654608 Ki = 15 nM T92072 C3D7FO 90654609 Ki = 20 nM T92072 C0TK1Z 90654610 Ki = 15 nM T92072 CM61SU 90654611 Ki = 6.7 nM T92072 CD1UL9 90654612 Ki = 14 nM T92072 CO2F1G 90654613 Ki = 3.1 nM T92072 C3KC0Q 90654614 Ki = 1.8 nM T92072 CEYO74 90654615 Ki = 2.5 nM T92072 CO6Q4L 90654616 EC50 = 4.6 nM T92072 CRD81F 90654617 EC50 = 9.5 nM T92072 CJZ1R8 90654618 Ki = 42 nM T92072 C8JX5C 90654619 Ki = 75 nM T92072 C9N3YR 90654620 Ki = 12 nM T92072 C6KG0A 90654621 Ki = 18 nM T92072 CV69KU 90654622 Ki = 11 nM T92072 C2DUS5 90654623 Ki = 2.4 nM T92072 C4O0EX 90654624 Ki = 6.3 nM T92072 C5CY9H 90654625 EC50 = 1.8 nM T92072 C73MVQ 90654626 Ki = 83 nM T92072 CT5KI6 90654627 Ki = 233 nM T92072 CRH37P 90663727 EC50 = 7.1 nM T92072 C8QN0D 90663728 EC50 = 8 nM T92072 CF7R0K 90663729 EC50 = 2.7 nM T92072 CA4H1M 90665174 Ki = 17 nM T92072 CXK5T1 90665312 Ki = 2960 nM T92072 CWPT08 90665313 Ki = 3030 nM T92072 CM78DN 90665314 Ki = 3560 nM T92072 C8DRF0 90665315 Ki > 10000 nM T92072 CJIO86 90665316 Ki > 10000 nM T92072 C02JAH 90665317 Ki > 10000 nM T92072 C2K1SF 90665318 Ki > 10000 nM T92072 C5BY8E 90667757 IC50 = 190.55 nM T92072 CH6KA8 90668272 Ki = 1170 nM T92072 CX9E1Z 90668273 Ki = 369 nM T92072 CYR6N5 90668274 Ki = 290 nM T92072 C73XJB 90668275 Ki = 3890 nM T92072 CFA6R0 90668276 Ki = 2960 nM T92072 CC1KY8 90668277 Ki > 5000 nM T92072 C0ROS7 101874280 Ki = 978 nM T92072 C1U9RW 101886899 Ki = 134.3 nM T92072 CPRH91 110171405 Ki = 250 nM T92072 CGBO72 118016229 Ki > 1000 nM T92072 C7AYV5 118540795 EC50 = 1430 nM T92072 CB74NK 118707149 Ki = 124 nM T92072 CFH85E 118707843 Ki = 385 nM T92072 COX73K 118707844 Ki = 57.1 nM T92072 CR13GS 118707845 Ki = 126 nM T92072 CS0WC2 118707846 Ki = 8990 nM T92072 C2A3FW 118707847 Ki = 296 nM T92072 CJ58XH 118707848 Ki = 365 nM T92072 CF78CL 118707849 Ki > 100000 nM T92072 C3K7UV 118707850 Ki = 317 nM T92072 C0UFO4 118707851 Ki = 322 nM T92072 CSW70B 118707852 Ki = 12700 nM T92072 CU9OE7 118707853 Ki > 100000 nM T92072 CGJW82 118707854 Ki > 100000 nM T92072 CUR32J 118707855 Ki = 162 nM T92072 C6O0RY 118707856 Ki = 613 nM T92072 CG10IH 118707857 Ki = 40 nM T92072 C9OHF2 118707858 Ki = 1150 nM T92072 CW72CL 118707859 Ki = 60.7 nM T92072 CL0U3C 118707860 Ki = 34.4 nM T92072 CL3NG5 118707861 Ki = 432 nM T92072 C9BSD0 118707862 Ki = 940 nM T92072 CDTJ73 118707863 Ki = 1340 nM T92072 CRDU39 118707864 Ki = 1250 nM T92072 C6Y5VQ 118707865 Ki = 932 nM T92072 CBO8V9 118707866 Ki = 866 nM T92072 C4CU6D 118707867 Ki = 1590 nM T92072 C4P5GH 118707868 Ki = 890 nM T92072 C9FKE5 118707869 Ki = 943 nM T92072 CNJ3Z4 118707870 Ki = 75.2 nM T92072 CXQY36 118707871 Ki = 231 nM T92072 C7SL4C 118707872 Ki = 176 nM T92072 CFR3Z1 118707873 Ki = 15600 nM T92072 C87ATB 118707874 Ki = 8860 nM T92072 C7HS6T 118707875 Ki = 13400 nM T92072 CXHQ82 118707876 Ki > 100000 nM T92072 CEQP75 118707877 Ki = 141 nM T92072 CY8OV1 118707878 Ki > 100000 nM T92072 CH5B6Y 118707879 Ki = 45.6 nM T92072 C3OJW0 118707880 Ki = 6510 nM T92072 CM5BE7 118707881 Ki > 100000 nM T92072 CHR1E9 118707882 Ki = 11900 nM T92072 CZW6U4 118707883 Ki = 10400 nM T92072 COR57B 118707884 Ki = 4490 nM T92072 C8C9TQ 118707885 Ki = 1780 nM T92072 C0NQ2O 118707886 Ki = 1110 nM T92072 CG68RH 118707887 Ki = 3790 nM T92072 C9CY3P 118707888 Ki = 2740 nM T92072 CNC81J 118707889 Ki = 5090 nM T92072 CM53PE 118707890 Ki = 2730 nM T92072 CL4B7K 118707891 Ki = 5760 nM T92072 CR20MO 118707892 Ki > 100000 nM T92072 C8WQ5E 118707893 Ki > 100000 nM T92072 CI6O9D 118707894 Ki > 100000 nM T92072 C28ABD 118707895 Ki = 30100 nM T92072 C56KNQ 118707896 Ki = 2450 nM T92072 C7LNI5 118708213 Ki = 64 nM T92072 C74OYF 118708214 Ki = 80 nM T92072 CJ9V4D 118708215 Ki = 90 nM T92072 C4KN7B 118708218 Ki = 75 nM T92072 CBG4I3 118708219 Ki = 375 nM T92072 CI53HJ 118708220 Ki = 90 nM T92072 CFOC02 118708225 Ki = 35 nM T92072 C1I8WJ 118708226 Ki = 155 nM T92072 C50PKS 118708228 Ki = 312 nM T92072 C1IFV4 118708231 Ki = 480 nM T92072 CGS1T2 118708232 Ki = 380 nM T92072 CM61FX 118708233 Ki = 420 nM T92072 CWU94Y 118708234 Ki = 5.3 nM T92072 CI29WS 118708235 Ki = 1.31 nM T92072 C2B0KW 118708236 Ki = 0.15 nM T92072 C0MXW8 118708237 Ki = 16 nM T92072 CX2B8P 118708238 Ki = 0.54 nM T92072 CQWJ06 118708239 Ki = 0.22 nM T92072 CL6P0G 118708240 Ki = 18 nM T92072 CYO73E 118714540 Ki = 500 nM T92072 CQZ6I2 118714543 Ki = 1890 nM T92072 CI76CX 118719026 Ki = 60 nM T92072 C9CJ3U 118721209 Ki = 1360 nM T92072 CEG12O 118721211 Ki = 4600 nM T92072 CPXH85 118721212 Ki = 1481 nM T92072 CR9D2E 118721213 Ki = 556 nM T92072 C91QXI 118721214 Ki = 565 nM T92072 CCL9T3 118721215 Ki = 1543 nM T92072 C3BP7M 118721216 Ki = 86 nM T92072 CZEL84 118721484 Ki = 127.4 nM T92072 CN4SK2 118721485 Ki = 1322 nM T92072 CYBW39 118721486 Ki = 2016 nM T92072 CSO42U 118723504 Ki = 172.5 nM T92072 CYQ9L7 118723505 Ki = 9.5 nM T92072 C0FO8N 118723506 Ki = 15.2 nM T92072 C1SN3J 118723507 Ki = 32.3 nM T92072 C8YUA2 118723508 Ki = 3.5 nM T92072 CZV1B8 118723509 Ki = 1.9 nM T92072 C7MD2E 118723510 Ki = 3.4 nM T92072 C85MGN 118723511 Ki = 1.4 nM T92072 CGAH24 118723512 Ki = 9.5 nM T92072 CQSA74 118723515 Ki = 12.9 nM T92072 C43KDA 118723517 Ki = 4.7 nM T92072 C6CKP5 118723518 Ki = 2.4 nM T92072 C2NBS8 118729966 Ki = 40800 nM T92072 CBH8G1 118729967 Ki > 30000 nM T92072 CA3IK7 118729968 Ki > 30000 nM T92072 CTL02Y 118729969 Ki > 10000 nM T92072 CGTA19 118729970 Ki = 7750 nM T92072 C8KX7U 118729971 Ki = 23500 nM T92072 CWJ48N 118729972 Ki > 100000 nM T92072 CU0W7P 118729973 Ki > 30000 nM T92072 CAS85G 118729974 Ki > 100000 nM T92072 CFX4R9 118729975 Ki = 32400 nM T92072 C6VC5A 118729976 Ki = 2380 nM T92072 CNG5S7 118729977 Ki > 10000 nM T92072 CD6GZ2 118729978 Ki > 30000 nM T92072 C03XWO 118729979 Ki > 30000 nM T92072 CZD98F 118729980 Ki > 30000 nM T92072 CE5Z7R 118729981 Ki = 14000 nM T92072 CBV0J4 118729982 Ki > 30000 nM T92072 C2A5CU 118729983 Ki = 19000 nM T92072 CM3S0N 118732278 Ki = 10200 nM T92072 CWQ54J 118732279 Ki = 8200 nM T92072 CQL0K7 118732280 Ki > 90000 nM T92072 CRK7H9 118732281 Ki = 40200 nM T92072 CK24DH 118732282 Ki = 8800 nM T92072 CP78KH 118732283 Ki = 900 nM T92072 CEO92J 118732284 Ki = 4000 nM T92072 CJ6YF9 118732285 Ki = 3500 nM T92072 CW62JS 118732286 Ki = 14000 nM T92072 CXW9U6 118732287 Ki > 100000 nM T92072 C06FRT 118732288 Ki > 100000 nM T92072 CR2CO8 118732289 Ki > 100000 nM T92072 C94GHE 118732290 Ki = 4300 nM T92072 COJ86X 118732291 Ki = 2800 nM T92072 C1KDT4 118732292 Ki > 100000 nM T92072 C7BO1N 118732293 Ki = 700 nM T92072 C4EFY5 118732294 Ki = 2700 nM T92072 CKV50L 118732295 Ki = 5100 nM T92072 CT3Q9E 118732296 Ki = 5000 nM T92072 CLRK73 118732297 Ki = 2500 nM T92072 CE85HO 118732298 Ki > 100000 nM T92072 C9Y6EK 118732299 Ki = 2600 nM T92072 CNJ1H0 118732300 Ki > 100000 nM T92072 CX6IN3 118732301 Ki > 100000 nM T92072 C4N6ZT 118732302 Ki > 100000 nM T92072 CDAZ14 118732303 Ki > 100000 nM T92072 CZ7TM6 118732304 Ki = 17700 nM T92072 CXZW46 118732305 Ki > 100000 nM T92072 CWX3P4 118732306 Ki = 5900 nM T92072 CXRT76 118732307 Ki = 600 nM T92072 CK0NS3 118732308 Ki = 2700 nM T92072 CRFJ71 118732309 Ki = 600 nM T92072 CT90VA 118732971 Ki = 0.919 nM T92072 CXM53U 118732972 Ki = 3.56 nM T92072 CF4G3P 118732973 Ki = 8.59 nM T92072 C3E2BJ 118732974 Ki = 0.682 nM T92072 C1U2FS 118732975 Ki = 0.311 nM T92072 C4YS5J 118732976 Ki = 0.453 nM T92072 CZ7QU0 118732977 Ki = 0.728 nM T92072 CHP93T 118732978 Ki = 1.23 nM T92072 CBT95M 118732979 Ki = 1.06 nM T92072 CZ3X0P 118732980 Ki = 0.432 nM T92072 CMDH59 118732981 Ki = 1.67 nM T92072 C7MZ9V 118732982 Ki = 2.39 nM T92072 CVS8R0 118734340 Ki > 10000 nM T92072 C91DBT 118734341 Ki > 10000 nM T92072 CV1JE8 118734342 Ki > 10000 nM T92072 C8AB7F 118734343 Ki > 10000 nM T92072 CLWV70 118734344 Ki > 10000 nM T92072 CP7SE9 118734345 Ki > 10000 nM T92072 CC0RE9 118734346 Ki > 10000 nM T92072 CV6X3F 118734347 Ki > 10000 nM T92072 CN8RI9 118734348 Ki > 10000 nM T92072 CEZ86B 118734349 Ki > 10000 nM T92072 C1QPJ3 118734350 Ki > 10000 nM T92072 CFH92R 118734351 Ki > 10000 nM T92072 CR8FT9 118734352 Ki > 10000 nM T92072 C8Y7QW 118734353 Ki > 10000 nM T92072 CR3Y1J 118734354 Ki > 10000 nM T92072 C5DL3X 118734355 Ki > 10000 nM T92072 CYB49C 118734356 Ki > 10000 nM T92072 CZE09N 118734357 Ki > 10000 nM T92072 CB7J1G 118734358 Ki > 10000 nM T92072 C79RHZ 118734359 Ki > 10000 nM T92072 CSAH95 118734360 Ki > 10000 nM T92072 C1CBG3 118734361 Ki > 10000 nM T92072 CN9S1Y 118734362 Ki > 10000 nM T92072 C5SQA1 118734363 Ki > 10000 nM T92072 CDVO89 118734364 Ki > 10000 nM T92072 CQ73IF 118734365 Ki > 10000 nM T92072 C43VAO 118734366 Ki > 10000 nM T92072 C4NQV6 118734367 Ki > 10000 nM T92072 CGF84C 118734368 Ki > 10000 nM T92072 C94UXF 118734369 Ki > 10000 nM T92072 CU0K8H 118734370 Ki = 147 nM T92072 CPY5O0 118734371 Ki = 243 nM T92072 CLI1V7 118734372 Ki = 8.12 nM T92072 CX08QC 118734373 Ki = 45 nM T92072 CD3BV5 118734374 Ki = 4.52 nM T92072 C58VBC 118734375 Ki > 10000 nM T92072 C0U1NA 118734376 Ki = 3.63 nM T92072 CZH87J 118734377 Ki = 75 nM T92072 C6R5EX 122178744 Ki > 1000 nM T92072 CH7X6K 122178745 Ki > 1000 nM T92072 C4EW6R 122178746 Ki > 1000 nM T92072 C0ORM6 122178747 Ki > 1000 nM T92072 C7WCK3 122178748 Ki > 1000 nM T92072 C0V6CM 122178749 Ki > 1000 nM T92072 C6CQP9 122178750 Ki > 1000 nM T92072 C3Z2FP 122178751 Ki > 1000 nM T92072 C1HA2V 122178752 Ki > 1000 nM T92072 C4LN2B 122178753 Ki > 1000 nM T92072 CC6X3Q 122178754 Ki > 1000 nM T92072 CA25IQ 122178755 Ki > 1000 nM T92072 CSKN51 122178756 Ki > 1000 nM T92072 C79XUV 122178757 Ki > 1000 nM T92072 C1MA9K 122182829 Ki = 3546 nM T92072 C06YKW 122182830 Ki = 1374 nM T92072 CT6L2Q 122182831 Ki = 2723 nM T92072 CZ45UW 122182832 Ki = 3087 nM T92072 CA1I5D 122182833 Ki = 8689 nM T92072 C9S2AG 122182834 Ki = 8024 nM T92072 C2R5TF 122182835 Ki = 1547 nM T92072 CQI46V 122182836 Ki = 8394 nM T92072 CDQ50Z 122182837 Ki = 4990 nM T92072 CU7NC1 122182838 Ki = 2411 nM T92072 CGJ4S6 122182839 Ki = 15920 nM T92072 CKR73I 122182840 Ki = 5847 nM T92072 CE7M1W 122182841 Ki = 4289 nM T92072 C8LIP2 122182842 Ki = 1920 nM T92072 CWE9G8 122182843 Ki = 1260 nM T92072 C6GTI8 122182881 Ki = 19780 nM T92072 C0D4IR 122182882 Ki = 19150 nM T92072 CG98FV 122188580 Ki = 2440 nM T92072 C2WK9L 122188584 Ki = 1350 nM T92072 CHEV48 122188585 Ki = 710 nM T92072 CKUJ38 122188742 EC50 = 2.9 nM T92072 CGN51R 122188744 Ki = 4.6 nM T92072 CNK9W4 122188745 Ki = 88 nM T92072 C7IM5S 122188746 Ki = 162 nM T92072 C5P7MB 122188747 Ki = 1.3 nM T92072 CI3PS0 122188748 EC50 = 1.9 nM T92072 C7LF5Y 122188749 EC50 = 1.9 nM T92072 CW0MC4 122188750 Ki = 2.3 nM T92072 CH3RC5 122188751 Ki = 3.8 nM T92072 CW58SR 122188752 Ki = 3.9 nM T92072 CZ63TJ 122188753 Ki = 12 nM T92072 CPA30H 122188754 Ki = 11 nM T92072 CV07OI 122188755 Ki = 11 nM T92072 CW3DC8 122188756 Ki = 9.3 nM T92072 C6S7RN 122188757 Ki = 19 nM T92072 CGC5Y6 122188758 EC50 = 7.6 nM T92072 C4WTB2 122188759 Ki = 24 nM T92072 CG7K1V 122188760 Ki = 53 nM T92072 C4CA3G 122444930 Ki = 337 nM T92072 CW58PY 122444937 Ki = 6300 nM T92072 C1G3QV 122444939 Ki = 213 nM T92072 CV9XW2 122444941 Ki = 132 nM T92072 CU2A5O 122444945 Ki = 6 nM T92072 CU65EJ 122444974 Ki = 20 nM T92072 C8QZN9 122444991 Ki = 1299 nM T92072 C5FMS9 122444992 Ki = 10 nM T92072 CW4LR8 122445001 Ki = 4743 nM T92072 C7WIN8 122445018 Ki = 135 nM T92072 CB5C8V 122485306 Ki = 57 nM T92072 CNQJ76 122485307 Ki = 213 nM T92072 C5M2OL 122485308 Ki = 84 nM T92072 CU8HB2 123131614 Ki > 10000 nM T92072 CX43WO 123131616 Ki > 10000 nM T92072 CKW26O 123131618 Ki = 9500 nM T92072 C1C5XE 127025020 Ki = 12 nM T92072 CBQY40 127025021 Ki = 31 nM T92072 CT2AL0 127025022 Ki = 346 nM T92072 C02MLK 127025023 Ki = 33 nM T92072 C9UQZ2 127025957 EC50 = 15848.93 nM T92072 C9OR6D 127025959 IC50 = 0.02951 nM T92072 CTL62C 127026187 Ki = 17620 nM T92072 CXG31M 127026188 Ki = 90 nM T92072 CFP01M 127026251 IC50 = 2.884 nM T92072 CS7TW8 127026252 IC50 = 37.15 nM T92072 C0MWD8 127026257 IC50 = 6.166 nM T92072 CLR2J7 127034153 IC50 = 29000 nM T92072 CH6L8J 127035004 Ki = 52 nM T92072 C2BM4D 127035624 Ki = 1180 nM T92072 CFJ95C 127035625 Ki = 946 nM T92072 CPY0S3 127035626 Ki = 311 nM T92072 CDWC03 127035803 Ki = 8960 nM T92072 CH41BT 127035804 Ki = 7150 nM T92072 C7AHR2 127035805 Ki = 1010 nM T92072 C92RXW 127035806 Ki = 676 nM T92072 CGD59Y 127035832 Ki = 361 nM T92072 CX29PN 127035833 Ki = 801 nM T92072 C4Y3XI 127035834 Ki = 306 nM T92072 CJM9Z1 127036437 Ki = 2570 nM T92072 CM63GQ 127036438 Ki = 3850 nM T92072 CA4E7T 127036562 Ki = 552 nM T92072 CLI39Z 127036563 Ki = 466 nM T92072 COD60T 127036564 Ki = 764 nM T92072 C59HYJ 127036640 Ki = 757 nM T92072 CJ52XA 127036641 Ki > 100000 nM T92072 CX9H5M 127036642 Ki > 100000 nM T92072 C4F2WP 127036740 Ki = 10500 nM T92072 C3QVM7 127036741 Ki = 24400 nM T92072 C3E7ZT 127036742 Ki = 7560 nM T92072 CGM30I 127036810 Ki = 63.9 nM T92072 CR7OT4 127036811 Ki = 2770 nM T92072 CR58OX 127036812 Ki > 100000 nM T92072 C65YKX 127036844 Ki = 784 nM T92072 CLCF05 127036845 Ki = 3080 nM T92072 C5K3MR 127036846 Ki > 100000 nM T92072 CB8HG0 127036933 Ki = 1450 nM T92072 C1MS0C 127036976 Ki = 1490 nM T92072 CQR43P 127036977 Ki > 100000 nM T92072 CMF9R6 127037424 Ki = 687 nM T92072 CY71PR 127037440 Ki = 400 nM T92072 C7LV5T 127038039 Ki = 1792 nM T92072 C2YT3C 127038355 Ki = 1940 nM T92072 C3CMX4 127038356 Ki = 358 nM T92072 CB63LH 127038545 Ki = 524 nM T92072 C3RV0U 127038566 Ki = 281 nM T92072 CB5F1H 127038752 Ki = 643 nM T92072 CN2R1H 127038755 Ki = 905 nM T92072 C86CAO 127038756 Ki = 1211 nM T92072 CHV76Y 127038890 Ki = 78 nM T92072 CB76CP 127038901 Ki = 40 nM T92072 CQ7SD5 127038919 Ki = 6037 nM T92072 C2OGT9 127040015 Ki = 90 nM T92072 CSU8G3 127040016 Ki = 103 nM T92072 CUD27T 127040064 Ki = 230 nM T92072 CFI5D8 127040304 Ki = 1910 nM T92072 CY4G8A 127040403 Ki = 19200 nM T92072 C9OG1N 127040410 Ki = 5620 nM T92072 CM5EQ3 127040561 Ki = 50 nM T92072 CA3HW8 127040562 Ki = 83 nM T92072 CVX0J9 127040563 Ki = 170 nM T92072 CNJ86G 127040564 Ki = 112 nM T92072 C64YFB 127041015 Ki = 24 nM T92072 C6G8HJ 127041016 Ki = 54 nM T92072 C3HEG8 127041017 Ki = 5.4 nM T92072 CWJ63T 127041018 Ki = 10000 nM T92072 CNL13K 127041019 Ki = 78 nM T92072 CN8YI1 127041044 Ki = 110 nM T92072 C7UT0I 127041279 Ki = 707 nM T92072 CXA76Q 127041420 Ki = 348 nM T92072 CK5ST2 127041635 Ki = 69 nM T92072 CI0BX5 127041636 Ki = 252 nM T92072 C15TGL 127041637 Ki = 748 nM T92072 CN5PD8 127041638 Ki = 6003 nM T92072 C2KNY6 127041935 Ki = 210 nM T92072 C0F5YR 127041936 Ki = 160 nM T92072 CQ4HV3 127042140 Ki = 116 nM T92072 CEN1Z7 127042141 Ki = 600 nM T92072 C8D4GN 127042408 Ki = 7600 nM T92072 CA1XD7 127042409 Ki = 138 nM T92072 C29QAL 127042479 Ki = 559 nM T92072 CXN90T 127042899 Ki = 160 nM T92072 CAZ71O 127042900 Ki = 120 nM T92072 C7ZOD5 127042993 Ki = 546 nM T92072 C10OFL 127042994 Ki = 2440 nM T92072 CGE9O0 127042995 Ki = 18600 nM T92072 CCV4W8 127042996 Ki = 2670 nM T92072 C4JR2S 127042997 Ki = 378 nM T92072 CD23GH 127043299 Ki = 974 nM T92072 CG8F3I 127043648 Ki = 7970 nM T92072 CZ5BA7 127043662 Ki = 2020 nM T92072 C1J3PR 127043818 Ki > 100000 nM T92072 C8V5EN 127043828 Ki = 1550 nM T92072 CMJL86 127044142 Ki = 2310 nM T92072 CYS6Z4 127044283 Ki = 629 nM T92072 CC6MG4 127044514 Ki > 100000 nM T92072 CW18JP 127044515 Ki = 399 nM T92072 C4O7WX 127044516 Ki > 30000 nM T92072 C3KQS4 127044517 Ki = 530 nM T92072 CE1A4H 127044518 Ki > 100000 nM T92072 CQJ71U 127044681 Ki > 30000 nM T92072 C7V4HX 127044785 Ki = 12600 nM T92072 CLXU52 127044795 Ki = 713 nM T92072 C5FC3T 127044855 Ki = 555 nM T92072 C53KHG 127045164 Ki = 17800 nM T92072 C5LC0U 127045165 Ki > 100000 nM T92072 CGS9B5 127045166 Ki > 100000 nM T92072 C8NV5Y 127045167 Ki = 539 nM T92072 C2R9PY 127045168 Ki = 1190 nM T92072 C0RMT7 127045169 Ki = 658 nM T92072 C7I3NV 127045170 Ki = 713 nM T92072 C6UK3Q 127045631 Ki = 1990 nM T92072 C8MT9L 127045699 Ki = 309 nM T92072 C02HYP 127045700 Ki = 252 nM T92072 C6VU1I 127045701 Ki = 60 nM T92072 C2GH3Q 127045815 Ki = 42 nM T92072 C4MQU2 127045909 Ki = 111 nM T92072 CQ1IB0 127045910 Ki = 65 nM T92072 CDHL50 127046050 Ki = 120 nM T92072 C3AJY8 127046301 Ki = 410 nM T92072 C80WYL 127046438 Ki = 159 nM T92072 CH8W3C 127046493 Ki = 98 nM T92072 COE1R5 127046494 Ki = 242 nM T92072 C72JQB 127046495 Ki = 136 nM T92072 C9OQ3P 127046496 Ki = 18 nM T92072 C8NI0K 127047720 Ki = 796 nM T92072 C34CWL 127047737 Ki = 49 nM T92072 CBW49E 127047803 Ki = 17 nM T92072 CW64PN 127047804 Ki = 103 nM T92072 CBF61Y 127047805 Ki = 52 nM T92072 C9MH4B 127047827 Ki = 5430 nM T92072 CC9U3O 127047927 Ki = 206 nM T92072 CV3K4L 127047929 Ki = 372 nM T92072 CNH42R 127051230 Ki = 5920 nM T92072 C97UBL 127051231 Ki > 100000 nM T92072 CZ9NH5 127051849 Ki > 100000 nM T92072 C4A3IX 127051850 Ki > 100000 nM T92072 C8ACT1 127051851 Ki > 100000 nM T92072 CY2B7M 127051852 Ki > 100000 nM T92072 CPN29G 127052152 Ki > 100000 nM T92072 CB6R7Z 127052168 Ki = 3360 nM T92072 C1TJ7B 132578491 Ki = 65.5 nM T92072 C5CKG0 132578492 Ki = 393 nM T92072 CVS8H1 132578493 Ki = 642 nM T92072 CKIA45 132933622 Ki = 6930 nM T92072 CA31YG 132938348 Ki = 480 nM T92072 C02UQE 132941757 Ki = 1200 nM T92072 CJ54MF 132991405 Ki = 3.54 nM T92072 C75XIA 132991406 Ki = 8.16 nM T92072 C3UC1T 134132667 Ki = 0.92 nM T92072 C2I7AE 134132684 Ki = 37 nM T92072 CHSK61 134133787 Ki = 221 nM T92072 CH53WN 134134340 Ki > 10000 nM T92072 CZ8HL0 134134668 Ki = 112 nM T92072 CT8B7O 134135300 Ki = 160 nM T92072 C6G4CW 134135745 Ki = 103 nM T92072 CTOK25 134137998 Ki = 205 nM T92072 C9A6KG 134138183 Ki = 76 nM T92072 CR38DS 134138275 Ki = 27 nM T92072 C7WPX1 134138322 Ki = 61 nM T92072 C8RVZ7 134138658 Ki = 12 nM T92072 CH0FX4 134138769 Ki = 144 nM T92072 CV38YZ 134138961 Ki = 163 nM T92072 CIAY28 134139825 Ki = 645 nM T92072 CBJW17 134140823 Ki = 54 nM T92072 CN9L1H 134141609 Ki = 104 nM T92072 C68AXD 134141831 Ki = 39 nM T92072 C2KSZ9 134142435 Ki = 8.51 nM T92072 C06AXV 134142495 IC50 = 2 nM T92072 C5ZAD2 134142611 Ki = 0.23 nM T92072 CR1YQ6 134142843 Ki = 6200 nM T92072 CSUL60 134142882 Ki = 30 nM T92072 CXFG86 134143159 Ki = 0.46 nM T92072 CJFV62 134143302 Ki = 397 nM T92072 C08RJA 134143536 Ki = 298 nM T92072 C5L9BD 134143752 Ki = 360 nM T92072 C2CQ8G 134143946 Ki = 38 nM T92072 CPFA07 134144066 Ki = 94 nM T92072 CBA6J2 134144170 Ki = 130 nM T92072 CWG9Q2 134144288 Ki = 0.55 nM T92072 C71PIY 134144970 Ki = 440 nM T92072 CC2YB7 134146826 Ki = 106 nM T92072 CPJN21 134147069 Ki = 180 nM T92072 C9T5ME 134147675 Ki = 1.76 nM T92072 C3L2PZ 134147788 Ki = 45 nM T92072 CRA5O4 134147994 Ki = 49 nM T92072 C4MDF2 134148336 Ki = 7.7 nM T92072 CY60SA 134148661 Ki = 144 nM T92072 CPI01N 134149255 Ki = 24 nM T92072 C0N8IS 134150832 Ki = 30 nM T92072 CGT32F 134150875 Ki = 14 nM T92072 CGXA08 134151211 Ki = 1.06 nM T92072 CNET28 134151346 Ki = 64 nM T92072 C8PT9W 134152052 Ki = 110 nM T92072 C73ISY 134152157 Ki = 117 nM T92072 CL2O6B 134152268 Ki = 59 nM T92072 CA29KP 134152503 Ki = 18 nM T92072 C1JK6T 134152846 Ki = 39 nM T92072 CK7M8Y 134153079 Ki = 1.4 nM T92072 CP41RT 134154065 Ki = 437 nM T92072 C7UOJ8 134156506 Ki = 104 nM T92072 C48WTR 134156643 Ki = 55 nM T92072 C20RNA 134157761 Ki = 41 nM T92072 C08ZQW 135404340 Ki = 35 nM T92072 C9WD5K 135405767 Ki > 1000 nM T92072 C61NZE 135409562 Ki = 1800 nM T92072 C2ATW9 135409793 Ki = 1310 nM T92072 CRVK68 135409825 Ki = 1900 nM T92072 C5T2ZE 135409960 Ki > 1000 nM T92072 C6G0HA 135416050 Ki > 1000 nM T92072 CI0HT3 135416055 Ki = 746 nM T92072 C1IEY0 135418256 IC50 = 1200 nM T92072 C0C5IU 135418454 Ki = 4 nM T92072 C0Z8RU 135421343 Ki > 1000 nM T92072 CW16MF 135421366 Ki = 1005 nM T92072 CUA67Z 135423046 Ki = 448 nM T92072 CT85YL 135428628 Ki = 60 nM T92072 CY9QI4 135428630 Ki = 35 nM T92072 C7P2ME 135428645 Ki = 22 nM T92072 C5OZ0L 135428653 Ki = 45 nM T92072 CI4Z3R 135430228 Ki = 810 nM T92072 CZA5F9 135436760 Ki > 1000 nM T92072 CJ6AW4 135437132 Ki = 140 nM T92072 C6HN3Z 135438480 Ki = 17 nM T92072 C4Y9OF 135439478 Ki = 251.19 nM T92072 CI4S7C 135440168 Ki = 955 nM T92072 CR9W5J 135440414 Ki > 1000 nM T92072 C1UNH9 135440428 Ki = 181 nM T92072 C3JA5S 135442119 Ki = 24 nM T92072 C5YUC2 135443302 Ki = 201 nM T92072 CO87CV 135443324 Ki > 1000 nM T92072 CWD8M7 135443353 Ki = 448 nM T92072 C4KLO0 135443378 Ki = 56 nM T92072 CG9IK2 135444614 Ki = 32 nM T92072 C9UCG0 135448286 Ki > 1000 nM T92072 C0B1XV 135454766 Ki > 1000 nM T92072 C28AWC 135463688 Ki = 501.19 nM T92072 C4DUN5 135464144 Ki = 398 nM T92072 CT4L7M 135465666 Ki = 204 nM T92072 CK47BF 135465712 Ki = 20 nM T92072 CU14JT 135465774 Ki = 3227 nM T92072 C1F5CA 135465776 Ki > 1000 nM T92072 C04XNV 135465778 Ki = 1993 nM T92072 CBV8I2 135465784 Ki > 1000 nM T92072 C7E2CQ 135465796 Ki = 2427 nM T92072 C0YZ3B 135470411 Ki > 1000 nM T92072 CW4V3S 135475677 Ki = 5.8 nM T92072 CPQ3J6 135477916 Ki > 1000 nM T92072 CK52RH 135483531 Ki = 168 nM T92072 CTU21N 135483619 Ki > 1000 nM T92072 CJ91TZ 135484407 IC50 = 3000 nM T92072 CI8R0L 135485985 Ki = 140 nM T92072 CE26MK 135486084 Ki = 548 nM T92072 CH0AR8 135486118 Ki = 467 nM T92072 C94GIL 135490950 Ki = 430 nM T92072 CVG5M0 135493238 Ki = 140 nM T92072 CCX3D7 135493268 Ki = 900 nM T92072 CF06CK 135493272 Ki > 1000 nM T92072 CS3OC8 135493279 Ki = 65 nM T92072 C9RS5H 135493280 Ki = 4481 nM T92072 CEI8W7 135493281 Ki = 520 nM T92072 C25QGD 135493285 Ki > 1000 nM T92072 CN10IO 135493286 Ki = 2410 nM T92072 C7O1NS 135493290 Ki > 1000 nM T92072 CV4X0H 135493292 Ki > 1000 nM T92072 C5OK7A 135499926 Ki = 100 nM T92072 CG3V6J 135501712 Ki = 23 nM T92072 CU8W5N 135508372 Ki > 1000 nM T92072 C28UOK 135509755 Ki = 3.1 nM T92072 CTB6R7 135515408 IC50 = 610 nM T92072 CFQ38U 135515507 Ki = 238 nM T92072 CCHU96 135516528 Ki = 42 nM T92072 C46YPU 135519330 Ki > 1000 nM T92072 CG64XS 135522362 Ki > 1000 nM T92072 C1E2ZK 135522363 Ki > 1000 nM T92072 C2CL8J 135522364 Ki = 1440 nM T92072 C2AHQ6 135522367 Ki = 566 nM T92072 CF9XI7 135522375 Ki > 1000 nM T92072 C4NG7Y 135522388 Ki = 150 nM T92072 C9A7QL 135522390 Ki > 1000 nM T92072 CUNG36 135522391 Ki > 1000 nM T92072 CFJ8P2 135525108 IC50 > 10000 nM T92072 C2WJI6 135529341 Ki > 1000 nM T92072 C7ARF8 135529362 Ki > 1000 nM T92072 C2V3CX 135529371 Ki = 850 nM T92072 CVXF23 135529372 Ki > 1000 nM T92072 CJ86ZY 135529373 Ki = 1898 nM T92072 CESZ83 135529396 Ki = 49 nM T92072 CJ4Y1H 135529398 Ki = 163 nM T92072 C2ET0M 135533291 Ki = 15 nM T92072 C8I2FM 135542466 Ki = 45 nM T92072 CU3F1O 135542558 Ki = 20 nM T92072 C51PIY 135543600 Ki = 413 nM T92072 CF3UQ4 135543624 Ki = 2.6 nM T92072 CKN9Y0 135543763 Ki = 6.1 nM T92072 C6WLJ3 135544018 IC50 > 10000 nM T92072 C1K5QE 135544028 IC50 > 10000 nM T92072 CR6X3F 135544059 IC50 > 10000 nM T92072 C38LZC 135545353 Ki > 1000 nM T92072 CI3LK7 135546224 IC50 = 1.5 nM T92072 C5Y9WX 135546648 Ki = 200 nM T92072 CESD69 135546649 Ki = 79 nM T92072 CUI90X 135546657 Ki > 1000 nM T92072 C5KX8N 135546658 Ki = 72 nM T92072 CNCD32 135566609 Ki = 0.1622 nM T92072 C8LBZ5 135624236 Ki = 3110 nM T92072 CV9P3G 135636727 Ki = 3019.95 nM T92072 CSO0H1 135646528 Ki = 776.25 nM T92072 C7KW6I 135678052 Ki > 1000 nM T92072 C6GI3C 135738646 IC50 = 27 nM T92072 C67BTG 135738649 IC50 > 38 nM T92072 CD6GS7 135738659 IC50 > 27 nM T92072 C6MHD7 135783184 Ki = 15.85 nM T92072 C62PTQ 135874413 Ki = 350 nM T92072 C87ZQJ 135874414 Ki > 1000 nM T92072 C9X1UL 135874415 Ki > 1000 nM T92072 CT40VW 135874416 Ki = 500 nM T92072 C1V9TY 135874420 Ki > 1000 nM T92072 C1T4GB 135874421 Ki > 1000 nM T92072 CFSX68 135874422 Ki > 1000 nM T92072 CNLH54 135874423 Ki > 1000 nM T92072 C2FK6J 135874424 Ki = 140 nM T92072 C04YTD 135874425 Ki > 1000 nM T92072 CIQ04D 135874427 Ki > 1000 nM T92072 C6TO4A 135874428 Ki = 480 nM T92072 CO0C5V 135874429 Ki = 675 nM T92072 C9JQ2C 135874430 Ki > 1000 nM T92072 CSOV01 135874431 Ki > 1000 nM T92072 C75TGS 135874432 Ki > 1000 nM T92072 C93GBH 135874433 Ki > 1000 nM T92072 CV7US0 135874434 Ki > 1000 nM T92072 CIVD34 135949027 Ki = 54 nM T92072 C01JXT 135949034 Ki = 61 nM T92072 C67IJL 135970557 Ki = 32359.37 nM T92072 C7JI8O 135976345 Ki = 15 nM T92072 CR47LG 135976467 EC50 = 100000 nM T92072 CLQ25B 135986772 Ki = 7244.36 nM T92072 C7R9LG 136002185 Ki > 1000 nM T92072 C3BV1J 136002186 Ki = 55 nM T92072 CSBL59 136002187 Ki > 1000 nM T92072 CGS18F 136002248 Ki = 2530 nM T92072 CUK9J5 136019511 Ki = 2525 nM T92072 CBZ1I4 136025838 Ki = 2510 nM T92072 CCS5F0 136025881 Ki = 3023 nM T92072 C2VZR6 136025990 Ki > 5000 nM T92072 CA17MI 136026025 Ki > 5000 nM T92072 C9SR2V 136026026 Ki > 5000 nM T92072 C6KNF2 136026027 Ki > 5000 nM T92072 CO90BT 136026133 Ki = 1078 nM T92072 CM3YH2 136026181 Ki > 5000 nM T92072 C38LUX 136036809 Ki > 1000 nM T92072 CEHF18 136042327 Ki > 1000 nM T92072 C4U7ZM 136042328 Ki = 155 nM T92072 CSR0Z3 136042329 Ki = 503 nM T92072 C9C2SF 136042330 Ki = 4558 nM T92072 C75CXE 136042331 Ki = 685 nM T92072 CS49WL 136042332 Ki = 4462 nM T92072 CQ2ZA9 136042333 Ki = 210 nM T92072 CON2J4 136042334 Ki = 734 nM T92072 C5VY2Z 136042335 Ki > 1000 nM T92072 CTEB06 136042336 Ki > 1000 nM T92072 CJW64L 136042337 Ki > 1000 nM T92072 C05QUF 136042338 Ki = 277 nM T92072 C0SX1K 136042339 Ki = 66 nM T92072 CQ37GX 136042340 Ki = 89 nM T92072 CF3BR5 136042341 Ki = 175 nM T92072 C75XRI 136042342 Ki = 304 nM T92072 CS7HM2 136042343 Ki = 65 nM T92072 C3S1WY 136042344 Ki > 1000 nM T92072 CR5H4M 136042345 Ki > 1000 nM T92072 C29YZE 136042346 Ki = 34 nM T92072 CAP1C6 136042347 Ki = 45 nM T92072 C5EX7D 136042348 Ki = 55 nM T92072 C4L7GE 136042349 Ki = 645 nM T92072 C9JM7Y 136042350 Ki = 150 nM T92072 CO15GM 136042351 Ki = 752 nM T92072 COEZ25 136042352 Ki = 280 nM T92072 CGX6H7 136042353 Ki = 576 nM T92072 C1W9XD 136042354 Ki = 736 nM T92072 CA6TI2 136042355 Ki = 222 nM T92072 CPUX51 136046111 Ki = 15 nM T92072 CJ75XH 136068601 Ki = 405 nM T92072 CL5B7U 136068602 Ki = 1200 nM T92072 CU6C4Z 136068688 Ki = 615 nM T92072 CSJE87 136068689 Ki = 545 nM T92072 C7SLK3 136068716 Ki = 2550 nM T92072 CZWP52 136068717 Ki = 2560 nM T92072 CDX2Q0 136068718 Ki > 5000 nM T92072 CY1RT3 136068719 Ki = 485 nM T92072 C2XW1I 136074047 Ki = 16.6 nM T92072 CI1PK7 136086896 Ki = 2040 nM T92072 C5HL7K 136086897 Ki = 1960 nM T92072 C6VLR1 136086898 Ki = 515 nM T92072 CL2E0U 136086899 Ki > 5000 nM T92072 C01GMB 136086900 Ki = 803 nM T92072 CA3X5T 136086901 Ki = 1530 nM T92072 CW49CH 136086902 Ki = 1900 nM T92072 C4F5WR 136086903 Ki = 1730 nM T92072 CS58QU 136086904 Ki > 5000 nM T92072 C4B1TU 136086905 Ki = 1680 nM T92072 CMOR91 136086906 Ki > 5000 nM T92072 C3HY9O 136086907 Ki > 5000 nM T92072 CWF2L1 136086908 Ki > 5000 nM T92072 CF8HV7 136183446 Ki = 122 nM T92072 C5EPJ2 136199393 Ki = 12 nM T92072 CF51IY 136228031 Ki > 10000 nM T92072 C5IX2C 136236319 Ki > 30000 nM T92072 CWL69G 136414902 Ki = 4200 nM T92072 CJY21N 137125272 Ki = 1.5 nM T92072 CGS61F 137553161 Ki = 8.96 nM T92072 CDZ07W 137631401 Ki = 37.5 nM T92072 CY61SG 137631471 Ki = 220 nM T92072 C9QS4J 137631671 Ki = 15 nM T92072 CE7LZ9 137632204 Ki = 420 nM T92072 CSM29H 137632333 Ki = 2000 nM T92072 CQ36UP 137632356 Ki > 30000 nM T92072 CH5F6G 137632488 Ki = 438 nM T92072 C92FIL 137632746 Ki > 30000 nM T92072 CFWO04 137632925 Ki = 14 nM T92072 CJ67UL 137633007 Ki = 8.9 nM T92072 C3WKU1 137633041 Ki = 91.1 nM T92072 C2AG4Y 137633276 Ki = 232 nM T92072 C9SYC5 137633560 Ki = 59.4 nM T92072 CZ2HV1 137633654 Ki = 4.35 nM T92072 CZC9A2 137633810 Ki = 1743 nM T92072 C8K7EM 137634052 EC50 = 257.04 nM T92072 C9YB3R 137634085 Ki = 1100 nM T92072 C71MVS 137634444 EC50 = 74.13 nM T92072 CRGN40 137635666 Ki = 247 nM T92072 CYL3X8 137636099 Ki = 1.79 nM T92072 CC9P6O 137636304 Ki = 2900 nM T92072 C01OZS 137636323 Ki = 698 nM T92072 CS1EO0 137636334 Ki = 45 nM T92072 CU9G8K 137636427 Ki = 1480 nM T92072 C9TUY7 137636552 Ki = 2060 nM T92072 CB6VZ3 137636630 Ki = 420 nM T92072 C6ABK1 137636769 Ki = 1880 nM T92072 C5P9LI 137637451 Ki = 115 nM T92072 C53RQW 137637667 Ki > 30000 nM T92072 CCTH80 137638080 Ki = 1.41 nM T92072 C91WNM 137638192 Ki = 210 nM T92072 CW4S1V 137638211 Ki > 30000 nM T92072 CQ8ZL2 137638623 Ki = 18 nM T92072 CZ9QX0 137639459 Ki = 2142 nM T92072 CTQ67J 137639588 EC50 = 1288.25 nM T92072 CS1K4G 137639818 Ki = 316 nM T92072 C0SC7L 137640093 Ki > 30000 nM T92072 C45FXO 137641603 Ki = 18.6 nM T92072 CG0DI3 137641858 EC50 = 77.62 nM T92072 C52XDH 137641906 Ki = 8.1 nM T92072 CFW9R5 137641990 Ki = 7.64 nM T92072 CV81KH 137642036 Ki = 0.438 nM T92072 C7QNC1 137642069 Ki = 12 nM T92072 CE4C5Y 137642150 Ki > 30000 nM T92072 CO94EX 137642153 Ki = 3.53 nM T92072 CB8L7K 137642940 Ki = 61.7 nM T92072 C7K9ZB 137642980 Ki > 30000 nM T92072 C76XKJ 137643150 Ki = 3704 nM T92072 CJQD73 137643164 EC50 = 35.48 nM T92072 CG46DW 137644190 Ki = 20 nM T92072 CPR72G 137644224 Ki = 247 nM T92072 C58QOM 137644249 Ki = 83.5 nM T92072 C4R0OC 137644481 Ki > 30000 nM T92072 CI7B3F 137645065 Ki = 24.6 nM T92072 CGLI82 137645223 Ki = 11.2 nM T92072 CF09IY 137645275 Ki > 30000 nM T92072 CY5IE9 137645551 Ki > 1000 nM T92072 CCW5R0 137645696 Ki = 1090 nM T92072 CDBT79 137645728 Ki = 13 nM T92072 C95UJV 137645798 Ki = 616 nM T92072 CJ20CU 137645935 Ki = 500 nM T92072 C8YN3Q 137646655 EC50 = 38.02 nM T92072 CER23T 137646828 EC50 = 56.23 nM T92072 CGL83H 137647102 Ki > 30000 nM T92072 CC0UF1 137647420 Ki = 0.95 nM T92072 CT91AP 137648111 Ki = 45 nM T92072 CCA7I4 137648143 Ki = 129 nM T92072 C1AIP8 137648928 Ki = 0.768 nM T92072 CS3DT1 137649083 EC50 = 134.9 nM T92072 C62KVF 137649307 Ki = 239 nM T92072 CWH89G 137649841 EC50 = 87.1 nM T92072 CIE03Y 137650221 Ki = 6.02 nM T92072 CBHR45 137650233 Ki = 524 nM T92072 C9W3PX 137650461 EC50 = 138.04 nM T92072 CIM50G 137650899 Ki = 10.7 nM T92072 CXCA79 137650918 EC50 = 29.51 nM T92072 C26YKP 137651319 Ki > 30000 nM T92072 CEAU34 137651531 Ki = 8.02 nM T92072 C13AMI 137651532 Ki > 30000 nM T92072 C9M7QE 137651747 Ki = 6.04 nM T92072 C52VBU 137651751 Ki = 311 nM T92072 C6Z1HJ 137651756 Ki = 1.89 nM T92072 C9G7TP 137652167 Ki = 3310 nM T92072 CVS93H 137652383 Ki = 139 nM T92072 C8T2HN 137652475 EC50 = 22.91 nM T92072 CJ24ZP 137653290 Ki = 47 nM T92072 CHYT41 137653409 EC50 = 34.67 nM T92072 CJ1R9K 137653588 Ki = 25.6 nM T92072 C4VJ5C 137654976 Ki = 25.2 nM T92072 C3AE6C 137655247 Ki = 570 nM T92072 CC94TW 137656049 Ki = 0.2 nM T92072 CA24YS 137656139 Ki = 491 nM T92072 CSJ3F9 137656764 Ki = 186 nM T92072 C28GAV 137656845 EC50 = 109.65 nM T92072 CJUE21 137656913 Ki = 3.5 nM T92072 C08KJH 137657382 Ki = 91.4 nM T92072 CH8PL9 137657570 Ki = 158 nM T92072 CW07LP 137657589 Ki = 440 nM T92072 CNTX97 137657841 Ki = 4.28 nM T92072 CJ8BC7 137657926 Ki = 0.454 nM T92072 CQ9BR1 137658051 Ki = 67 nM T92072 C4XSN0 137658330 Ki = 180 nM T92072 CBC31H 137658387 Ki > 30000 nM T92072 CH9A8M 137658761 Ki = 1.87 nM T92072 CRH98I 137658892 Ki = 143 nM T92072 CV7UE3 137659204 Ki = 1000 nM T92072 CY67UM 137659236 Ki > 30000 nM T92072 CO6B8M 137659407 Ki = 156 nM T92072 C7VNS4 137659441 Ki = 3.73 nM T92072 CT23EA 137659930 Ki = 44 nM T92072 C1NZL8 137659963 Ki > 30000 nM T92072 CIDG46 137660466 Ki = 21.1 nM T92072 C3Y2IZ 137661132 Ki = 2.71 nM T92072 CFUM75 137661322 Ki = 59.4 nM T92072 C26LVX 137661505 EC50 = 93.33 nM T92072 C1DL4J 137661670 Ki = 17.6 nM T92072 COM9G6 137661811 Ki > 30000 nM T92072 CD1Z9C 137661874 Ki = 41.8 nM T92072 CT26DO 137662145 Ki = 5740 nM T92072 CP02WU 139030524 EC50 = 1.43 nM T92072 CU3PW1 139248507 Ki > 1000 nM T92072 CT1H6B 139248508 Ki > 1000 nM T92072 CUIN96 139248509 Ki > 1000 nM T92072 CW74BD 141536950 Ki = 12500 nM T92072 C6SUZ3 143294251 Ki = 603 nM T92072 CN2LX1 144852560 Ki = 1120 nM T92072 CBV2L5 145436760 Ki = 12.5 nM T92072 CK15TH 145436761 Ki = 25 nM T92072 C6KOB8 145436762 Ki = 5.24 nM T92072 CM7J2Q 145436763 Ki = 2.61 nM T92072 CSQL37 145436764 Ki = 8.12 nM T92072 CNP52A 145436765 Ki = 4.92 nM T92072 C6OFP7 145436766 Ki = 28 nM T92072 CSQ8U5 145436767 Ki = 7.12 nM T92072 C4PZ5S 145436769 Ki = 38 nM T92072 CI75YJ 145949481 Ki = 71 nM T92072 C2GVM4 145954098 Ki = 73 nM T92072 CQ9G0K 145954398 Ki = 29 nM T92072 C3RU6S 145954471 Ki = 70 nM T92072 CZX79R 145954995 Ki = 54000 nM T92072 CC0OX1 145958464 Ki = 17.3 nM T92072 CH7G6S 145960536 Ki = 333 nM T92072 C9PT5Q 145960667 Ki = 140 nM T92072 C3BY8E 145960746 Ki = 253 nM T92072 CWSM81 145960813 Ki = 43 nM T92072 CA9TS3 145960852 Ki = 3535 nM T92072 C5D6AI 145960873 Ki = 121 nM T92072 C62JCL 145960933 Ki = 1000 nM T92072 CQ6G3T 145961023 Ki = 724 nM T92072 CQN69Z 145961145 Ki = 113 nM T92072 CRBY29 145961339 Ki = 547 nM T92072 C0WBV6 145961509 Ki = 2665 nM T92072 C02OQR 145961748 Ki = 112 nM T92072 C1O0GQ 145961937 Ki = 338 nM T92072 CCB0Y2 145961997 Ki = 195 nM T92072 CT8UO0 145962202 Ki = 32 nM T92072 C3M7ZN 145962234 Ki = 485 nM T92072 CVA89T 145962310 Ki = 242 nM T92072 CD6X5O 145962355 Ki = 10.2 nM T92072 C86APL 145962364 Ki = 531 nM T92072 CH5DS7 145962529 Ki = 92 nM T92072 CJH4A7 145962653 Ki = 782 nM T92072 C4NXC1 145962657 Ki > 10000 nM T92072 CN0AG6 145962770 Ki = 1153 nM T92072 CPB32D 145962986 Ki = 3721 nM T92072 C6EFM0 145963225 Ki = 912 nM T92072 C9UYI6 145963230 Ki = 37 nM T92072 CQH82E 145963272 Ki = 2874 nM T92072 C5MD4S 145963661 Ki = 281 nM T92072 CLT8E9 145964522 Ki = 483 nM T92072 C86XTA 145965011 Ki = 66 nM T92072 C01PVB 145965471 Ki = 8.2 nM T92072 CYZ05R 145967103 Ki = 21 nM T92072 C4CN1A 145967785 Ki = 140 nM T92072 C1ER6I 145967791 Ki = 714 nM T92072 CJ81MI 145970314 Ki = 872 nM T92072 C8J7FL 145971923 Ki = 47 nM T92072 CNU0Q9 145972065 Ki = 338 nM T92072 CZJA45 145972655 Ki = 37 nM T92072 CR89KO 145972761 Ki = 44 nM T92072 CE23KG 145973077 Ki = 235 nM T92072 CV9OM2 145973260 Ki = 1700 nM T92072 CBT7E9 145973326 Ki > 10000 nM T92072 CJH7D0 145974358 Ki = 83 nM T92072 CZ9WQ0 145975577 Ki = 536 nM T92072 CKMZ02 145975919 Ki = 345 nM T92072 C9TLO2 145976032 Ki = 552 nM T92072 CI2HN1 145977111 Ki >= 10000 nM T92072 CM1R0J 145977114 Ki = 104 nM T92072 C8W0MQ 145978569 Ki = 67 nM T92072 C5SZN2 145979632 Ki = 12100 nM T92072 C43NUZ 145980000 Ki = 1910 nM T92072 COK2V5 145980546 Ki = 250 nM T92072 CO3Y8B 145980553 Ki = 37500 nM T92072 CP92RY 145980571 Ki = 6710 nM T92072 C7NJH2 145980712 Ki = 102 nM T92072 CMFW02 145980971 Ki = 26.4 nM T92072 CDM63O 145981315 Ki = 93.9 nM T92072 CHQ73C 145981492 Ki = 58.7 nM T92072 CA9R1X 145981583 Ki = 23.4 nM T92072 CX02DQ 145981864 Ki = 190 nM T92072 CNTY13 145982075 Ki = 34.3 nM T92072 CAI53J 145982270 Ki = 313 nM T92072 CHSJ14 145982423 Ki = 2340 nM T92072 C8RT4W 145982945 Ki = 177 nM T92072 C9CG6I 145984161 Ki > 100000 nM T92072 CUM74P 145984609 Ki = 21900 nM T92072 C9VDN3 145985635 Ki = 33300 nM T92072 C19BNU 145986670 Ki = 39200 nM T92072 CQ9AK0 145987082 Ki = 48.3 nM T92072 CJ70FS 145987226 Ki = 744 nM T92072 C05IZF 145987813 Ki > 100000 nM T92072 CGV37C 145987819 Ki = 51 nM T92072 C0AF1D 145988094 Ki = 130 nM T92072 CD01TO 145988590 Ki = 6500 nM T92072 C3O1MT 145988709 Ki = 4190 nM T92072 CMD74V 145988733 Ki = 172 nM T92072 CV53QZ 145988884 Ki = 1300 nM T92072 CEM2L0 145989440 Ki = 122 nM T92072 CVS17Y 145989611 Ki = 3850 nM T92072 CB9GL1 145989764 Ki = 19700 nM T92072 C4I1EY 145990207 Ki > 100000 nM T92072 C98GKM 145990252 Ki = 1680 nM T92072 CZP5T3 145990301 Ki = 4100 nM T92072 CJ0A5L 145990511 Ki = 19800 nM T92072 CHV8C9 145990554 Ki = 38 nM T92072 C3H2ZP 145990725 Ki = 348 nM T92072 CJ30YT 145990769 Ki = 41 nM T92072 CC4BW2 145990800 Ki = 7.7 nM T92072 C2Y8PA 145990926 Ki = 33500 nM T92072 CV5XO6 145991048 Ki = 246 nM T92072 C6ZYL7 145991283 Ki = 1360 nM T92072 C9YO2T 145991303 Ki = 2080 nM T92072 CN7A1X 145991427 Ki = 48600 nM T92072 CUP48Y 145991545 Ki = 79.7 nM T92072 C8QT3X 145991607 Ki = 25400 nM T92072 C7K5ZQ 145991651 Ki > 100000 nM T92072 C8SI9A 145991749 Ki = 277 nM T92072 C2CB3J 145991827 Ki = 137 nM T92072 C3QHT6 145992189 Ki = 216 nM T92072 C1MU4D 145992652 Ki = 46.6 nM T92072 CB85AS 145992677 Ki = 3670 nM T92072 C94OJE 145992790 Ki = 556 nM T92072 C7B3FY 145992928 Ki = 73.1 nM T92072 C47DOA 145993092 Ki > 100000 nM T92072 CZOR31 145993511 Ki = 55.2 nM T92072 CQ93KE 145993540 Ki = 2390 nM T92072 C6A3RN 145993941 Ki = 119 nM T92072 CO69HC 145994068 Ki > 100000 nM T92072 C72SMW 145994175 Ki > 100000 nM T92072 CE07TR 145994259 Ki = 28.3 nM T92072 C5LXC4 153605593 Ki = 2.14 nM T92072 CZ53NG 153605599 Ki = 17.8 nM T92072 C4W8PK 155413621 Ki > 10000 nM T92072 C2CG8J 155510487 Ki = 2870 nM T92072 C14XVK 155510489 Ki = 69 nM T92072 CEXH54 155511332 Ki = 2 nM T92072 CD52TC 155511687 Ki = 935 nM T92072 CPMN94 155511844 Ki = 40 nM T92072 CCD9N1 155512086 Ki = 22.7 nM T92072 CTV8R1 155512151 Ki = 63.4 nM T92072 C4FA0V 155512157 Ki = 2.9 nM T92072 CM5ZA9 155512438 Ki = 205 nM T92072 CTP3K1 155512498 Ki = 2290 nM T92072 CX96QM 155512576 Ki > 100000 nM T92072 CLUF91 155513199 Ki = 9502 nM T92072 CV35ZN 155513505 Ki = 4.9 nM T92072 CGS27D 155513515 Ki = 45.9 nM T92072 CU67HI 155513890 Ki = 1050 nM T92072 CV20JC 155513938 Ki = 5.1 nM T92072 CP7UX3 155513958 Ki = 794.33 nM T92072 CUB2C9 155514153 Ki = 93 nM T92072 C38LUS 155514209 Ki = 391.7 nM T92072 CST9B5 155514281 Ki > 10000 nM T92072 CR85FY 155514357 Ki = 1770 nM T92072 CQ7GR6 155514463 Ki = 67 nM T92072 CF04MH 155514522 Ki = 2.5 nM T92072 CGIT15 155514690 Ki > 10000 nM T92072 CRF2B1 155514696 Ki = 1.42 nM T92072 CN8E1J 155514860 Ki = 795 nM T92072 CP6C5S 155514957 Ki > 1000 nM T92072 CLJ7Y3 155515226 Ki = 5520 nM T92072 C9NJT8 155515787 Ki = 2511.89 nM T92072 CNV02U 155516016 Ki >= 10000 nM T92072 CT18NO 155516071 Ki = 479.2 nM T92072 CLX4D7 155516277 Ki = 419 nM T92072 CR59VH 155517789 Ki = 32 nM T92072 C0CR9Q 155518147 Ki > 1000 nM T92072 CR5VO9 155518410 Ki = 79.43 nM T92072 C2PM8H 155518462 Ki = 4.5 nM T92072 CR40UE 155518944 Ki = 12 nM T92072 CP74IJ 155519148 Ki = 28 nM T92072 C0EAY4 155519375 Ki = 742 nM T92072 CX1MO3 155519551 Ki = 2.71 nM T92072 C5YDE2 155519621 Ki = 687 nM T92072 CEY82J 155519727 Ki > 100000 nM T92072 C5NTJ8 155519776 Ki = 58.5 nM T92072 C72OJY 155519986 Ki = 378.6 nM T92072 C8N1CQ 155520115 Ki = 8.4 nM T92072 CXS1T4 155520635 Ki > 10000 nM T92072 CZ1S5N 155520662 Ki = 28.9 nM T92072 CPL4Q7 155520955 Ki = 175.5 nM T92072 C6A4UH 155521103 Ki = 594 nM T92072 CS2GJ8 155521355 Ki = 2275 nM T92072 C25KBM 155521478 Ki > 30000 nM T92072 C1LH7J 155521488 Ki = 4.7 nM T92072 CYW7Q0 155521543 Ki > 1000 nM T92072 CXD9G0 155521637 Ki = 50.12 nM T92072 CW29KY 155521694 Ki = 262.7 nM T92072 CHTX98 155522541 Ki > 1000 nM T92072 CSBN54 155522680 Ki = 7536 nM T92072 CGJ0W4 155522875 Ki = 1359 nM T92072 CBW5G4 155522899 Ki = 47.7 nM T92072 C0S4EM 155522991 Ki = 208 nM T92072 C3SJ9B 155523748 Ki = 34 nM T92072 CK8RS0 155523968 Ki = 113 nM T92072 C4ZIH2 155524032 Ki > 1000 nM T92072 CMLS87 155524113 Ki = 4.6 nM T92072 C8E3HR 155524516 Ki = 334 nM T92072 CYSK39 155525038 Ki > 30000 nM T92072 CZX2N4 155525050 Ki > 1000 nM T92072 CN1C6R 155525265 Ki = 29.7 nM T92072 C8QIF6 155525396 Ki = 10 nM T92072 C78DHT 155525494 Ki = 4.5 nM T92072 CR6A7N 155525747 Ki = 62.3 nM T92072 CT24MQ 155526752 Ki = 9.8 nM T92072 CBAK91 155527112 Ki = 1220 nM T92072 C5CO8R 155527265 Ki = 341 nM T92072 CS9U0T 155527740 Ki = 21.3 nM T92072 C15MXV 155527829 Ki = 37 nM T92072 C3BEX2 155527968 Ki = 630.96 nM T92072 C3KA0S 155528136 Ki > 1000 nM T92072 CAR75Z 155528717 Ki > 1000 nM T92072 CZ53GQ 155528757 Ki = 2550 nM T92072 CXM9W5 155529088 Ki = 15848.93 nM T92072 CZWH28 155529694 Ki = 13 nM T92072 CZ9YC8 155529872 Ki = 535 nM T92072 CZF94H 155530202 Ki = 398.11 nM T92072 CVE30Z 155530257 Ki > 1000 nM T92072 CS2BT0 155530292 Ki = 1.22 nM T92072 CQT8O2 155530381 Ki > 1000 nM T92072 C78JZY 155530514 Ki = 928 nM T92072 CN87UW 155530961 Ki = 1100 nM T92072 CNVU03 155531548 Ki = 175.9 nM T92072 C3XQ9S 155531570 Ki = 288.7 nM T92072 C4A3DX 155531727 Ki > 1000 nM T92072 C14GCE 155531842 Ki = 186 nM T92072 CQI01K 155531990 Ki > 1000 nM T92072 C7A9BH 155532173 Ki = 33 nM T92072 C21MLU 155532274 Ki > 1000 nM T92072 CVI21H 155532514 Ki > 1000 nM T92072 C86SCT 155532773 Ki = 13670 nM T92072 CJH8R0 155532913 Ki = 22 nM T92072 CQ96YB 155532918 Ki = 4070 nM T92072 C9EU2D 155533104 Ki > 100000 nM T92072 CY0H3U 155533272 Ki = 1200 nM T92072 CY8O6B 155533349 Ki = 778 nM T92072 C03YFW 155533388 Ki = 8 nM T92072 C9TLW2 155533451 Ki = 158.49 nM T92072 CCG1K2 155533519 Ki = 60 nM T92072 C7E5OP 155533880 Ki = 5110 nM T92072 CH54UR 155534188 Ki = 8480 nM T92072 CW8FN0 155534473 Ki = 1472 nM T92072 C9QV4W 155534659 Ki = 102.7 nM T92072 C4NU8B 155534836 Ki > 1000 nM T92072 COT9U8 155535203 Ki = 961 nM T92072 C9ZK5A 155535230 Ki > 10000 nM T92072 CRQW57 155535452 Ki = 19 nM T92072 C67VZK 155535458 Ki = 10400 nM T92072 C38WUG 155536405 Ki = 243 nM T92072 CIUS98 155536619 Ki = 495 nM T92072 CH6E1O 155536745 Ki = 1036 nM T92072 C6Q1EM 155536934 Ki = 2500 nM T92072 C8ZG7F 155537023 Ki = 3520 nM T92072 C3P8VK 155537874 Ki > 10000 nM T92072 CW75BA 155538492 Ki = 649 nM T92072 C8BHN2 155540525 Ki = 55 nM T92072 CF6ZE5 155540615 Ki = 73 nM T92072 C3P1ZT 155540839 Ki > 1000 nM T92072 C2L9TS 155540948 Ki > 1000 nM T92072 C4KDO9 155541051 Ki = 2.72 nM T92072 C42QAK 155541530 Ki = 240 nM T92072 C2HX6J 155541790 Ki = 13 nM T92072 C9H5VC 155541975 Ki > 100000 nM T92072 CQ1FY8 155542311 Ki = 1.18 nM T92072 CMEW36 155542520 Ki = 1.02 nM T92072 CGY1J4 155542588 Ki = 7100 nM T92072 CCV87Q 155542600 Ki > 1000 nM T92072 C0BFX9 155542720 Ki > 1000 nM T92072 C06OKY 155542884 Ki = 82 nM T92072 CR8A7D 155543424 Ki = 9142 nM T92072 C3XDT7 155543719 Ki = 148 nM T92072 CMT60C 155543832 Ki = 120 nM T92072 C2DNQ0 155543871 Ki > 60000 nM T92072 C1QAZ9 155544096 Ki = 2580 nM T92072 CR0EV6 155544177 Ki > 100000 nM T92072 CQ9Z2P 155545386 Ki = 51 nM T92072 CJS87Q 155545399 Ki = 4850 nM T92072 C5Y4BH 155545414 Ki = 791 nM T92072 C5HU6A 155545585 Ki = 560 nM T92072 C45CUJ 155545762 Ki > 1000 nM T92072 CZ49CM 155545843 Ki = 2710 nM T92072 CM5ZN0 155545870 Ki > 30000 nM T92072 C2NKO5 155545904 Ki = 265 nM T92072 C3B0SI 155546100 Ki = 28 nM T92072 C95ICF 155546118 Ki = 7820 nM T92072 C4BHE8 155546183 Ki > 1000 nM T92072 CL1T9K 155546550 Ki = 42.6 nM T92072 CHC2O5 155547064 Ki = 4.1 nM T92072 C1VHM5 155547186 Ki > 100000 nM T92072 CQE30Y 155547305 Ki = 12200 nM T92072 CXAV84 155547390 Ki = 89 nM T92072 C6XJ0D 155547715 Ki = 324 nM T92072 C35WAK 155548264 Ki > 1000 nM T92072 C39GTQ 155548778 Ki = 224.6 nM T92072 CY1XJ0 155548779 Ki > 100000 nM T92072 C82STM 155549033 Ki = 125.89 nM T92072 C3NE6F 155549264 Ki > 1000 nM T92072 CY5U1J 155549967 Ki > 10000 nM T92072 CY7Q9N 155550159 Ki > 1000 nM T92072 C2IU1J 155550532 Ki > 1000 nM T92072 C6J5EX 155550807 Ki = 236 nM T92072 CN2I3H 155550832 Ki > 100000 nM T92072 CT7MV5 155551482 Ki > 10000 nM T92072 C41JXM 155551530 Ki > 10000 nM T92072 C4LN3W 155551750 Ki = 1010 nM T92072 CI41QF 155552117 Ki = 7.61 nM T92072 CA29GP 155552390 Ki = 77.7 nM T92072 CJ82KN 155552405 Ki > 1000 nM T92072 CF0W4K 155552683 Ki = 1750 nM T92072 CIQH30 155552719 Ki > 1000 nM T92072 CPN79B 155553292 Ki = 82 nM T92072 CX4P7S 155553385 Ki > 100000 nM T92072 CD42WK 155553510 Ki = 59 nM T92072 CNK6Z9 155553575 Ki > 1000 nM T92072 CY08CH 155553600 Ki = 6944 nM T92072 CG1CF2 155553962 Ki = 70 nM T92072 CU1ZE5 155554091 Ki = 1.32 nM T92072 CFW01A 155554317 Ki > 30000 nM T92072 CPXQ16 155554464 Ki = 0.98 nM T92072 C57MKC 155555241 Ki > 1000 nM T92072 CWCN91 155555408 Ki = 2.6 nM T92072 CVDO87 155555721 Ki > 1000 nM T92072 CN38KO 155555854 Ki = 8560 nM T92072 CL3IB5 155555868 Ki = 1660 nM T92072 CJ73SL 155556032 Ki > 1000 nM T92072 CDR63F 155556134 Ki = 1461 nM T92072 CYB6T5 155556258 Ki = 10400 nM T92072 CV9P2M 155556457 Ki = 492 nM T92072 CBS89O 155556618 Ki = 32.7 nM T92072 C7M1VE 155556836 Ki > 100000 nM T92072 CGF0H2 155556884 Ki > 1000 nM T92072 CV21NW 155557226 Ki = 553 nM T92072 C2F1JY 155557284 Ki = 40800 nM T92072 CDYO34 155557387 Ki = 44.8 nM T92072 CJ16GB 155557960 Ki > 1000 nM T92072 C7FUQ6 155558172 Ki = 65 nM T92072 C0W7AL 155558312 Ki = 3880 nM T92072 CDMC47 155558350 Ki = 108.5 nM T92072 C8Z2TC 155558489 Ki = 265 nM T92072 CYX8T1 155558921 Ki = 0.51 nM T92072 CIAE48 155558941 Ki > 30000 nM T92072 CVS4T6 155559056 Ki > 100000 nM T92072 CDZX46 155559070 Ki = 2.11 nM T92072 C5EC8U 155559408 Ki = 2680 nM T92072 CP87XK 155559423 Ki = 396 nM T92072 C0RWG1 155559434 Ki = 630.96 nM T92072 CQM64H 155559636 Ki = 33.5 nM T92072 CV5PC7 155559963 Ki = 7856 nM T92072 C34ORN 155560261 Ki > 100000 nM T92072 C8B7CG 155560391 Ki > 1000 nM T92072 C73XYW 155560510 Ki = 492 nM T92072 CN93BY 155560649 Ki = 57 nM T92072 C5KY7D 155561141 Ki = 326 nM T92072 CGD7R4 155561189 Ki = 190 nM T92072 C49XPN 155561350 Ki = 398.11 nM T92072 CQ2L0P 155561909 Ki > 10000 nM T92072 CKG56Z 155562044 Ki = 1750 nM T92072 CXUN73 155562096 Ki = 4.12 nM T92072 C6EN2B 155562182 Ki = 356 nM T92072 C5X9FM 155562751 Ki > 10000 nM T92072 CM46KC 155563177 Ki > 1000 nM T92072 CQ19VC 155563189 Ki > 1000 nM T92072 C4N9GU 155563428 Ki = 73.8 nM T92072 CJZO26 155563438 Ki > 100000 nM T92072 CE2V5Y 155564179 Ki > 1000 nM T92072 C8TL6J 155564465 Ki = 364 nM T92072 CHJ5Q8 155564753 Ki > 30000 nM T92072 CFNC10 155565326 Ki = 17.6 nM T92072 C0UFM3 155565444 Ki = 632 nM T92072 C8N3PQ 155565636 Ki = 651 nM T92072 CB14WJ 155565911 Ki >= 1000 nM T92072 C6DQ1K 155566338 Ki = 23.6 nM T92072 C0VUO9 155566764 Ki > 1000 nM T92072 CN8RL3 155567003 Ki > 30000 nM T92072 CPW8M5 155567457 Ki = 1490 nM T92072 C5KNM6 155569051 Ki = 1440 nM T92072 C7Q9WY 11395785 Ki = 1.2 nM T92072 C4EBT3 16109359 EC50 = 3.388 nM T92072 CQT04G 16109362 EC50 = 5.129 nM T92072 C19DJN 16109368 EC50 = 0.6918 nM T92072 CJZ23T 44333154 Ki > 10000 nM T92072 CIU68M 44333155 Ki > 10000 nM T92072 CV8BQ7 44333404 Ki > 10000 nM T92072 C30UYD 44333842 Ki = 3476 nM T92072 CCK07J 44333843 Ki = 6350 nM T92072 C90IQB 46905977 Ki = 3920 nM T92072 D00ASZ 16204411 Ki = 218 nM T92072 D00CJJ 12016636 Ki = 12000 nM T92072 D00CVD 252716 Ki > 10000 nM T92072 D00GNW 16109429 Ki = 0.87 nM T92072 D00GQI 11313151 Ki = 11.1 nM T92072 D00HYS 18507264 Ki = 3.3 nM T92072 D00JMT 210332 Ki > 10000 nM T92072 D00JWA 46880333 Ki = 358 nM T92072 D00MFV 44572293 Ki = 34000 nM T92072 D00MPA 9834240 Ki = 4951 nM T92072 D00NFW 16109432 Ki = 2.4 nM T92072 D00NYG 2303947 Ki = 10.8 nM T92072 D00OFN 44420099 Ki = 67 nM T92072 D00WFU 11381543 Ki = 8.87 nM T92072 D00YOM 15557795 Ki = 4180 nM T92072 D00YXE 11652061 Ki > 10000 nM T92072 D01CQU 5139184 Ki = 157 nM T92072 D01EHP 4401 Ki = 1081 nM T92072 D01MOQ 13155595 Ki = 50.12 nM T92072 D01NHH 16109434 Ki = 5.5 nM T92072 D01PGY 10045125 Ki = 97 nM T92072 D01QBK 44572356 Ki = 4600 nM T92072 D01QYQ 6603931 Ki = 210 nM T92072 D01VEU 44300688 Ki = 1280 nM T92072 D01VXC 11278089 Ki = 31.3 nM T92072 D01VXP 16115754 Ki = 25 nM T92072 D01WNA 5248753 Ki = 280 nM T92072 D01WXR 12253310 Ki = 483 nM T92072 D02BGA 9877796 Ki = 0.4 nM T92072 D02EAO 11243768 Ki = 2730 nM T92072 D02FLH 16109427 Ki = 2.5 nM T92072 D02HOL 11849871 Ki = 1100 nM T92072 D02HYT 11438116 Ki = 9.5 nM T92072 D02HZJ 11245073 Ki = 671 nM T92072 D02JMR 16202727 Ki = 145 nM T92072 D02NBB 44449695 Ki = 3920 nM T92072 D02RBK 9904551 Ki = 6700 nM T92072 D02TEW 10754789 Ki = 45 nM T92072 D02WTN 11404772 Ki = 109 nM T92072 D02XPR 73124 Ki > 100000 nM T92072 D02ZZQ 44567454 Ki > 100000 nM T92072 D03FVK 16115753 Ki = 1190 nM T92072 D03HBG 16203543 Ki = 443 nM T92072 D03JFX 7 Ki = 7400 nM T92072 D03KLO 9815374 Ki = 101 nM T92072 D03NVE 10226014 Ki > 6000 nM T92072 D03POP 44420681 Ki = 1210 nM T92072 D03RFA 657378 EC50 = 0.19 nM T92072 D04AGC 18511481 Ki = 16500 nM T92072 D04DVT 126079 Ki = 175 nM T92072 D04JIR 69689 Ki = 12000 nM T92072 D04LZN 44572409 Ki = 2200 nM T92072 D04PJO 10612371 Ki = 21 nM T92072 D04SDD 44436081 EC50 > 3000 nM T92072 D04TTP 127993 Ki = 7370 nM T92072 D04WHE 247436 Ki = 9400 nM T92072 D04XLX 44449523 Ki = 60 nM T92072 D04YUM 75929 Ki > 100000 nM T92072 D04ZTH 2817024 Ki = 43 nM T92072 D05KEF 44418996 Ki = 0.55 nM T92072 D05MCK 6105572 Ki = 0.1585 nM T92072 D05SYY 10402581 Ki = 0.7943 nM T92072 D05TFM 44449741 Ki = 3205 nM T92072 D05XGF 44186581 Ki = 2240 nM T92072 D05ZRR 9836155 Ki = 4027 nM T92072 D05ZUX 44207909 Ki >= 1000 nM T92072 D06FNT 10247610 Ki > 10000 nM T92072 D06GOE 135465785 Ki > 1000 nM T92072 D06GTI 135416058 Ki > 1000 nM T92072 D06KYP 44572292 Ki = 830 nM T92072 D06NQD 695136 Ki = 274 nM T92072 D06QRI 10378184 Ki = 0.631 nM T92072 D06RCT 16203429 Ki = 148 nM T92072 D06SGU 11774068 Ki > 6000 nM T92072 D06TSQ 135494270 Ki = 23 nM T92072 D06ZWQ 4962866 Ki = 203 nM T92072 D07DGH 11450364 Ki = 27.6 nM T92072 D07DOE 44447542 Ki = 21 nM T92072 D07FGB 11709210 Ki = 235 nM T92072 D07FZA 135522368 Ki = 700 nM T92072 D07HXL 122028 EC50 = 1700 nM T92072 D07IPZ 11740439 Ki = 95 nM T92072 D07YKU 44449258 Ki = 1466 nM T92072 D08AJS 135407706 Ki = 3336 nM T92072 D08AXT 44449696 Ki = 5765 nM T92072 D08CIY 11424684 Ki = 56 nM T92072 D08EBT 10981286 Ki = 327 nM T92072 D08EZI 11739042 Ki = 14.8 nM T92072 D08FOT 5311479 Ki > 10000 nM T92072 D08HBH 11359018 Ki = 17.6 nM T92072 D08INY 619020 Ki = 25.2 nM T92072 D08JUQ 11652153 Ki = 4 nM T92072 D08JYX 11743895 Ki = 1280 nM T92072 D08LZN 11450197 Ki = 3000 nM T92072 D08RGW 44403594 Ki = 8720 nM T92072 D08SJF 44403591 Ki > 10000 nM T92072 D09HAM 10491577 Ki = 659 nM T92072 D09IRV 11523232 Ki = 0.73 nM T92072 D09KUY 12431921 Ki = 1000 nM T92072 D09RKX 135433658 Ki = 1640 nM T92072 D09UDF 44449257 Ki = 2041 nM T92072 D09VOP 16203665 Ki = 1820 nM T92072 D09VRX 11521761 Ki = 8000 nM T92072 D0A0VT 44572291 Ki > 100000 nM T92072 D0A4MK 135489238 Ki = 300 nM T92072 D0A5KG 16094571 Ki = 230 nM T92072 D0A6IO 5310960 Ki = 1100 nM T92072 D0A6JX 452612 Ki = 8700 nM T92072 D0A9BZ 11605883 Ki = 2067 nM T92072 D0AI8F 12016633 Ki = 1000 nM T92072 D0B0QW 10389852 Ki = 730 nM T92072 D0B0TX 44572355 Ki = 4900 nM T92072 D0B2NE 44598833 Ki = 32800 nM T92072 D0B3UE 12852 Ki = 10000 nM T92072 D0B8RQ 11427528 Ki = 2.22 nM T92072 D0BC7P 3355253 Ki = 22 nM T92072 D0C1PS 12486289 Ki > 100000 nM T92072 D0C2UJ 8974 Ki = 1.39 nM T92072 D0C3ID 11314132 Ki = 309 nM T92072 D0CB9B 9813424 Ki = 675 nM T92072 D0CX7N 44572471 Ki = 1000 nM T92072 D0D3WR 44401938 Ki = 3324 nM T92072 D0D4NS 11536096 Ki > 10000 nM T92072 D0DB7A 414707 Ki = 4300 nM T92072 D0E2FV 309375 Ki > 100000 nM T92072 D0E4LB 16115752 Ki = 282 nM T92072 D0E4UT 13789211 Ki > 100000 nM T92072 D0E5QE 25113696 Ki > 100000 nM T92072 D0E7YE 11462181 Ki = 21 nM T92072 D0E8RA 2773172 Ki = 16000 nM T92072 D0F4EN 11470612 Ki > 1000 nM T92072 D0F4XB 2817165 Ki = 12 nM T92072 D0F8CV 5462471 Ki > 100000 nM T92072 D0FF6S 16038374 IC50 > 10000 nM T92072 D0G5ZF 10318664 Ki = 437 nM T92072 D0G6BI 16203542 Ki = 253 nM T92072 D0G6VT 16202726 Ki = 350 nM T92072 D0H2VA 9884349 Ki = 11 nM T92072 D0H9BP 5697 Ki = 6.82 nM T92072 D0H9EY 10475082 Ki = 3.3 nM T92072 D0HK5B 9798914 Ki = 350 nM T92072 D0I1IW 16203539 Ki = 150 nM T92072 D0I2EQ 16109426 Ki = 14 nM T92072 D0I7HL 14842885 Ki = 960 nM T92072 D0IG5E 44582613 Ki = 1.56 nM T92072 D0J3TY 10588437 Ki = 12 nM T92072 D0J4EZ 135443359 Ki > 1000 nM T92072 D0J4SW 10731097 Ki = 29 nM T92072 D0J6ME 9964781 Ki = 917 nM T92072 D0JJ6T 10021483 Ki = 0.54 nM T92072 D0K0OT 1329 Ki = 0.47 nM T92072 D0K5WC 44567438 Ki > 100000 nM T92072 D0K6ZA 5311041 Ki = 37 nM T92072 D0K8ZZ 448222 EC50 = 0.12 nM T92072 D0KJ3H 16203431 Ki = 197 nM T92072 D0KM0Y 10423637 Ki = 12 nM T92072 D0KT3L 10454501 Ki = 2790 nM T92072 D0L0VU 135484064 Ki = 200 nM T92072 D0L2MN 11529627 Ki = 27 nM T92072 D0L4TY 11301995 Ki = 25.1 nM T92072 D0L6YI 16203540 Ki = 358 nM T92072 D0L7DL 11610347 Ki = 36 nM T92072 D0LP5V 11536936 Ki = 0.82 nM T92072 D0M3CG 93205 Ki = 2 nM T92072 D0N0OE 46229111 Ki = 5000 nM T92072 D0N1PT 11500124 Ki = 350 nM T92072 D0N1QO 10320311 Ki = 1870 nM T92072 D0N1QP 16109423 Ki = 1.2 nM T92072 D0N2DP 11484484 Ki = 4470 nM T92072 D0N2VO 668105 Ki = 14 nM T92072 D0N8RM 242652 Ki = 29000 nM T92072 D0N9WG 11234532 Ki = 368 nM T92072 D0NF3E 11565524 Ki > 10000 nM T92072 D0O0FP 9860294 Ki = 71.8 nM T92072 D0O4KI 9834769 Ki = 388 nM T92072 D0O6NS 81457 Ki = 33000 nM T92072 D0OR5V 414708 Ki > 100000 nM T92072 D0OX0V 11688103 Ki = 0.5 nM T92072 D0P0BV 16202841 Ki = 310 nM T92072 D0P5ZE 11771279 Ki > 10000 nM T92072 D0P7FK 743242 Ki = 5.8 nM T92072 D0P8MK 44572469 Ki = 1500 nM T92072 D0PU1R 12431922 Ki > 10000 nM T92072 D0PU6F 11658819 Ki = 50 nM T92072 D0Q1RD 16202725 Ki = 130 nM T92072 D0Q3LM 16115477 Ki = 22 nM T92072 D0Q5HW 9801709 Ki = 1380 nM T92072 D0Q6KO 1942 Ki = 29000 nM T92072 D0Q6WX 2690 Ki = 4.4 nM T92072 D0Q9GL 135443367 Ki = 250 nM T92072 D0QD3O 619024 Ki = 17.7 nM T92072 D0QN4U 16202728 Ki = 210 nM T92072 D0QN5I 9964493 Ki = 479 nM T92072 D0R1XY 123807 IC50 = 0.5012 nM T92072 D0R4LZ 11536774 Ki = 32 nM T92072 D0R8OK 822296 Ki = 570 nM T92072 D0RZ2M 11572592 Ki = 4.1 nM T92072 D0S4JI 20262 Ki > 100000 nM T92072 D0S5XP 44572408 Ki = 8400 nM T92072 D0S6QA 11608719 Ki = 3200 nM T92072 D0T2RY 9948320 Ki >= 1000 nM T92072 D0T7GG 16109430 Ki = 0.62 nM T92072 D0TC7N 9953255 Ki = 560 nM T92072 D0TU7I 5353365 Ki > 10000 nM T92072 D0U8KW 46203501 EC50 = 177.83 nM T92072 D0UM6O 44449565 Ki = 615 nM T92072 D0V7MX 247678 Ki > 100000 nM T92072 D0V8MD 1922 IC50 = 1340 nM T92072 D0V9EE 24950370 Ki = 28 nM T92072 D0W1PF 16109428 Ki = 0.61 nM T92072 D0W3MT 11565892 Ki = 4.4 nM T92072 D0W5CZ 21976428 Ki = 2765 nM T92072 D0W6FC 44572473 Ki = 2900 nM T92072 D0W6TG 44186666 Ki > 10000 nM T92072 D0W8RB 44572357 Ki = 4900 nM T92072 D0WI4D 11617054 Ki = 0.29 nM T92072 D0WN3O 11290921 Ki = 27.1 nM T92072 D0X5PJ 135529391 Ki > 1000 nM T92072 D0Y5TL 5372720 Ki > 100000 nM T92072 D0Y5WQ 44185871 Ki > 10000 nM T92072 D0Y6HQ 16115478 Ki = 255 nM T92072 D0Y7AV 44449709 Ki = 10000 nM T92072 D0Y8EU 393595 Ki = 231 nM T92072 D0Y8LD 135529386 Ki > 1000 nM T92072 D0Y8SB 4355631 IC50 = 5300 nM T92072 D0Y9WZ 44583036 Ki = 68 nM T92072 D0Z1WY 44447548 Ki = 15.5 nM T92072 D0Z2QM 23562742 Ki = 20000 nM T92072 D0Z3BT 11462102 Ki = 8.75 nM T92072 D0Z3XC 11185362 Ki = 31.2 nM T92072 D0Z3YY 11392960 Ki = 3.7 nM T92072 D0Z7BC 44442164 Ki = 50 nM T92072 D0Z8NC 16109435 Ki = 0.9 nM T92072 D0Z8VU 44572295 Ki = 3100 nM T92072 D0ZF8N 11196622 Ki > 1000 nM T92072 D0ZV1T 11371386 Ki = 6.35 nM T92072 D0ZW9L 11150373 Ki = 8.6 nM T92557 CHS5T6 291557 IC50 = 45000 nM T92557 C6MPQ5 1473632 IC50 = 650000 nM T92557 C1XME6 6914573 IC50 = 230 nM T92557 CR6U4D 9580781 IC50 = 150000 nM T92557 C4CU8X 10157845 IC50 = 12900 nM T92557 CQ84VN 10199773 IC50 = 3200 nM T92557 C85XKJ 10222293 IC50 = 2500 nM T92557 C9P7JF 10269359 IC50 = 4200 nM T92557 C58NDH 10270253 IC50 = 2350 nM T92557 C8HJ9A 10272344 IC50 > 35000 nM T92557 CZ7R5G 10291281 IC50 = 12800 nM T92557 C98VXF 10293153 IC50 = 2800 nM T92557 CK3X8L 24180049 IC50 = 36000 nM T92557 CLD84G 44410488 IC50 = 51000 nM T92557 C3K2GM 44410492 IC50 = 1200 nM T92557 CBLP98 44410493 IC50 = 5700 nM T92557 CG07UX 44410495 IC50 = 800 nM T92557 C2FY1X 44410581 IC50 = 37200 nM T92557 CWU6D2 44410692 IC50 = 15000 nM T92557 CH6FW7 44410693 IC50 = 56800 nM T92557 C1R6JP 44410694 IC50 = 1160 nM T92557 CB7MP1 44410703 IC50 = 33300 nM T92557 CM01XR 56671820 IC50 = 15000 nM T92557 CY8MK2 56671821 IC50 = 360000 nM T92557 CPM14W 56675216 IC50 = 105000 nM T92557 CD3I4T 78319104 IC50 = 251.19 nM T92557 C2UCV5 118988431 IC50 = 3981.07 nM T92557 C3YPW8 122190023 IC50 = 63.1 nM T92557 CE6YK2 127043627 IC50 = 1258.93 nM T92557 D0AW6C 9879950 IC50 = 18300 nM T92557 D0W0FI 9967156 IC50 = 13300 nM T63359 C19ORL 11273626 IC50 = 5800 nM T63359 CFWM26 16049809 IC50 = 9800 nM T63359 CQ6HG2 16078804 IC50 = 54000 nM T63359 C4W9CO 16078805 IC50 = 42000 nM T63359 CO8W4C 16078806 IC50 = 54000 nM T63359 CLA43G 16078807 IC50 = 8600 nM T63359 CKSO26 16078808 IC50 = 8700 nM T63359 CSQ95P 16078809 IC50 = 4800 nM T63359 C4K8NF 16078810 IC50 = 4800 nM T63359 C6FX4U 16078811 IC50 = 13000 nM T63359 CA3J1G 16078812 IC50 = 10000 nM T63359 C9EBG4 16078813 IC50 = 4500 nM T63359 C9I4NR 16078814 IC50 = 5400 nM T63359 C3FA6X 16078815 IC50 = 6100 nM T63359 C6QXC5 16078816 IC50 = 5800 nM T63359 C2G4PU 16078817 IC50 = 5900 nM T63359 CC8RE2 16078818 IC50 = 40000 nM T63359 CJD94F 16078819 IC50 = 8100 nM T63359 CPD0Y2 16078820 IC50 = 11000 nM T63359 CY5D6A 44400303 IC50 > 50000 nM T63359 C6H1UC 44400324 IC50 = 7200 nM T63359 CC0W8S 44400490 IC50 = 7200 nM T63359 CQR0O7 44400556 IC50 > 50000 nM T63359 CF51RI 44400564 IC50 = 49000 nM T63359 COW7U2 44400587 IC50 = 20000 nM T63359 CSU7V5 44417242 IC50 = 5600 nM T63359 CI7B8O 44417248 IC50 = 17600 nM T63359 CCLN67 44417249 IC50 < 6200 nM T63359 C2XG3C 44417256 IC50 > 52000 nM T63359 C63PZU 44417262 IC50 = 21900 nM T63359 CN43GD 44417274 IC50 = 5500 nM T63359 C2N1HO 44417275 IC50 > 44000 nM T63359 CL0ZH6 44417284 IC50 < 6200 nM T63359 CW8FV0 44417291 IC50 = 5900 nM T63359 C8Y0ZN 44417294 IC50 = 12200 nM T63359 CMD9H5 44417295 IC50 < 6200 nM T63359 CO38IN 44417301 IC50 < 6200 nM T63359 C0WP3I 44417306 IC50 = 13100 nM T63359 CNH9Y3 44417307 IC50 = 9600 nM T63359 CRXF52 54679840 IC50 = 3 ug.mL-1 T63359 CXKE26 54682555 IC50 = 10 ug.mL-1 T63359 C8UN1J 54712725 IC50 = 5 ug.mL-1 T63359 C39MDC 54728582 IC50 = 8 ug.mL-1 T63359 CHC41J 54728583 IC50 = 3 ug.mL-1 T63359 CXQ08D 54728584 IC50 = 2 ug.mL-1 T63359 CPU1Q7 54728585 IC50 > 25 ug.mL-1 T63359 C8OAV0 54728586 IC50 = 1 ug.mL-1 T63359 C3Q4ZU 54728587 IC50 > 25 ug.mL-1 T63359 CYF20S 54728588 IC50 = 9 ug.mL-1 T63359 C70FLC 54728589 IC50 > 25 ug.mL-1 T63359 C26FBM 54728590 IC50 = 4 ug.mL-1 T63359 C0SXV7 54728591 IC50 = 10 ug.mL-1 T63359 CK0BJ9 54728592 IC50 > 25 ug.mL-1 T63359 CWS12N 54728593 IC50 = 10 ug.mL-1 T63359 CONQ08 54728594 IC50 = 2 ug.mL-1 T63359 C1Q3YH 54728595 IC50 > 25 ug.mL-1 T63359 C69NOJ 54728596 IC50 = 2 ug.mL-1 T63359 C9CGU2 54728597 IC50 = 1 ug.mL-1 T63359 CGXT73 54728598 IC50 = 6 ug.mL-1 T63359 CA19RH 54728599 IC50 = 12 ug.mL-1 T63359 C2G9XV 54728600 IC50 = 1 ug.mL-1 T63359 C5LYS9 54728604 IC50 = 3 ug.mL-1 T63359 CAWP39 54728605 IC50 > 25 ug.mL-1 T63359 COFR80 54728606 IC50 = 1 ug.mL-1 T63359 CW0L3M 54728607 IC50 = 11 ug.mL-1 T63359 C4U1RG 54728608 IC50 = 3 ug.mL-1 T63359 CB4QF3 135967825 IC50 > 55000 nM T72841 D07KSG 2733526 IC50 = 200 nM T72841 D08QMX 5757 EC50 = 5.9 nM T72841 D0JO7Y 104741 IC50 = 2 nM T72841 D0L4FS 5280961 IC50 = 10 nM T72841 CDN6F7 9985556 IC50 = 440 nM T72841 CUZ01R 11156792 IC50 = 750 nM T72841 C9CME0 11166839 IC50 = 1400 nM T72841 C9Y2NB 11179472 IC50 = 2600 nM T72841 C21VGK 11191381 IC50 = 1700 nM T72841 C4AVT7 11191582 IC50 = 1500 nM T72841 C0GZC2 11203882 IC50 = 2000 nM T72841 C37TYX 11260667 IC50 = 920 nM T72841 CR4X0F 11328702 IC50 = 3300 nM T72841 CRX32S 11352626 IC50 = 1800 nM T72841 CTSV17 11375459 IC50 = 2200 nM T72841 CW9K1H 11376935 IC50 = 500 nM T72841 CH9SR7 11420191 IC50 = 2000 nM T72841 CI16OE 11421901 IC50 > 10000 nM T72841 CE2TX0 11431360 IC50 = 1800 nM T72841 C5YLD8 11432134 IC50 = 800 nM T72841 CG48HJ 11432898 IC50 = 540 nM T72841 C2BAO3 11582785 IC50 = 470 nM T72841 C9OZI1 11668937 IC50 = 470 nM T72841 C0G5MI 11719412 IC50 = 57 nM T72841 C9BC0L 16732000 Ki > 10000 nM T72841 C5KGC6 24825442 IC50 = 700 nM T72841 CC53XL 24860583 Ki > 2300 nM T72841 CX3I6O 25008509 IC50 = 16 nM T72841 CU2B6A 25008510 IC50 = 70 nM T72841 CBL1J3 25008680 IC50 = 240 nM T72841 C0C3ZJ 25008854 IC50 = 165 nM T72841 CX8N1E 25009027 IC50 = 13 nM T72841 C30HJO 25009028 IC50 = 62 nM T72841 C6FL9N 25009030 IC50 = 720 nM T72841 C3C6HW 25009031 IC50 = 140 nM T72841 CUM01J 25009191 IC50 = 540 nM T72841 C8PR6D 44397271 IC50 = 2300 nM T72841 CN9L7G 46916268 IC50 = 33 nM T72841 CF59JY 49891022 IC50 = 3600 nM T72841 CD07PE 51050929 IC50 = 720 nM T72841 C0G1BK 51050930 IC50 = 800 nM T72841 CZ84BA 51050931 IC50 = 350 nM T72841 CITQ74 51051023 IC50 = 730 nM T72841 CKH39D 51051024 IC50 = 1800 nM T72841 CB3YF8 51051025 IC50 = 2600 nM T72841 CTS4G2 51051026 IC50 = 290 nM T72841 C52JPE 51051027 IC50 = 1100 nM T72841 CC43AH 51051028 IC50 = 280 nM T72841 C7D1SN 51051119 IC50 = 1000 nM T72841 CZ3WJ4 51051120 IC50 = 2400 nM T72841 C70BHM 51051121 IC50 = 500 nM T72841 CA14XO 51051122 IC50 = 47 nM T72841 CZ5A4S 51051123 IC50 = 80 nM T72841 CC40ZN 51051124 IC50 = 36 nM T72841 C1RP3V 51051125 IC50 = 68 nM T72841 C0MP7H 51051230 IC50 = 890 nM T72841 C01HPF 51051231 IC50 = 640 nM T72841 CZ3FY9 51051232 IC50 = 220 nM T72841 CB4R3E 51051233 IC50 = 1300 nM T72841 C8U6SC 51051234 IC50 = 1000 nM T72841 CM7BY6 53385590 IC50 = 14000 nM T72841 C5ZX4B 54597874 IC50 = 23 nM T72841 C7GAK5 54674240 IC50 = 22 nM T72841 CY9IT6 54674251 IC50 = 15 nM T72841 CF7XA0 54674257 IC50 = 34 nM T72841 CIE32B 58530397 IC50 = 43 nM T72841 C92CPO 58530407 IC50 = 580 nM T72841 C4TFB2 58530409 IC50 = 16 nM T72841 C45BUQ 58530416 IC50 = 19 nM T72841 CE0BC6 58530433 IC50 = 9 nM T72841 C0QUC6 58530436 IC50 = 5 nM T72841 C8K1VO 58530485 IC50 = 13 nM T72841 C9K4DS 58530524 IC50 = 23 nM T72841 C0LF1C 58530563 IC50 = 28 nM T72841 CHLQ30 58530589 IC50 = 18 nM T72841 CCB84G 58530630 IC50 = 26 nM T72841 CP56MI 58530705 IC50 = 9 nM T72841 CK5TZ7 58530717 IC50 = 24 nM T72841 CKBS71 58530720 IC50 = 8 nM T72841 CHI20F 58530748 IC50 = 46 nM T72841 CCR83N 58530759 IC50 = 8 nM T72841 C7F5TX 58530789 IC50 = 25 nM T72841 CS9J8N 58530798 IC50 = 23 nM T72841 CLZ65G 58530888 IC50 = 19 nM T72841 CQH91G 58530912 IC50 = 54 nM T72841 C8H6NR 58530923 IC50 = 12 nM T72841 CID86K 58530931 IC50 = 8 nM T72841 C2PV6W 58530954 IC50 = 17 nM T72841 CB54WI 71605373 IC50 = 50 nM T72841 CV9N4F 71605540 IC50 = 50 nM T72841 C56KSX 71605541 IC50 = 96.5 nM T72841 CYW9V0 71605542 IC50 = 126.4 nM T72841 CM07WE 71605543 IC50 = 28.3 nM T72841 C7EIS1 71605704 IC50 = 637.8 nM T72841 C7NBI8 71605705 IC50 = 175.7 nM T72841 C3LD2H 71605706 IC50 = 100 nM T72841 C3J5UW 71605707 IC50 = 24.4 nM T72841 CX85NI 71681512 IC50 = 1590 nM T72841 CG79WE 71681513 IC50 = 1440 nM T72841 COY32Z 71681514 IC50 = 390 nM T72841 C1K5GO 71681515 IC50 = 900 nM T72841 C67JYR 71681516 IC50 = 890 nM T72841 C5PD9X 71681677 IC50 = 9530 nM T72841 CL0CO1 71681678 IC50 > 50000 nM T72841 CAQ07F 71681679 IC50 = 2070 nM T72841 C1XN3R 71681680 IC50 = 41 nM T72841 CNR2Y6 71681681 IC50 = 310 nM T72841 CE52BO 71681682 IC50 = 160 nM T72841 CBT4E6 71681683 IC50 = 1540 nM T72841 C7K8WF 71681684 IC50 = 3950 nM T72841 CX5F9H 71681838 IC50 = 21 nM T72841 CMAZ46 71681839 IC50 = 200 nM T72841 CR0D5K 71681840 IC50 = 2170 nM T72841 C56INM 71681841 IC50 = 15890 nM T72841 C84BDM 71681842 IC50 = 430 nM T72841 CHV56D 71681843 IC50 = 94 nM T72841 CO7EB8 71681844 IC50 = 650 nM T72841 CV69XI 71681845 IC50 = 1740 nM T72841 C2CI3G 71682010 IC50 > 50000 nM T72841 C8T2RB 71682011 IC50 = 72 nM T72841 CV56YB 71682012 IC50 = 100 nM T72841 C5QD4B 71682013 IC50 = 1040 nM T72841 CJ09DS 71682014 IC50 > 50000 nM T72841 C6JMY1 71682015 IC50 > 50000 nM T72841 CFS9J7 71682016 IC50 > 50000 nM T72841 CGQF87 86659644 IC50 = 23 nM T72841 CE17QA 86659645 IC50 = 25 nM T72841 CN8P1G 90307845 IC50 = 15 nM T72841 C4J5EA 91799292 IC50 = 8 nM T72841 CFQ6P8 122182191 IC50 = 21080 nM T72841 C2URL4 134134246 IC50 > 10000 nM T72841 CD7NA5 134138492 IC50 > 10000 nM T72841 CP04WC 134144077 IC50 = 8100 nM T72841 CYG76M 134150509 IC50 > 10000 nM T72841 C89SMK 134152807 IC50 > 10000 nM T72841 C1O0IW 134153257 IC50 > 10000 nM T72841 C0Z4OD 134155524 IC50 > 10000 nM T72841 C58OUX 134155994 IC50 = 8010 nM T72841 CI2OM9 135399711 IC50 = 144 nM T72841 CH2K3S 135424843 IC50 = 150 nM T72841 C67LAW 135427962 IC50 = 65 nM T72841 C30QWY 135430315 IC50 = 28 nM T72841 CB3XM0 135438509 IC50 = 86 nM T72841 CVBN04 135446024 IC50 = 319 nM T72841 CB5P0O 135461031 IC50 = 160 nM T72841 CYJ96L 135508068 IC50 = 94 nM T72841 CA3F6J 135508229 IC50 = 6.1 nM T72841 C1BJU2 135546507 EC50 = 1000 nM T72841 CNXJ86 137628681 IC50 > 10000 nM T72841 CK5F9L 137631419 IC50 = 80 nM T72841 CL7B2E 137633187 IC50 = 170 nM T72841 CUT05L 137633831 IC50 = 770 nM T72841 CDR9F7 137641916 IC50 = 210 nM T72841 CAB21C 137644849 IC50 = 280 nM T72841 CF21JL 137648953 IC50 = 490 nM T72841 C6Q8XV 137650814 IC50 = 570 nM T72841 C9F3VU 137652631 IC50 = 170 nM T72841 C5Q3TI 137655175 IC50 = 22 nM T72841 CW3ZO6 137657402 IC50 = 390 nM T72841 CX4FK5 137657442 IC50 = 650 nM T72841 CUB6Q0 137661569 IC50 > 1000 nM T72841 C8NO5Z 139291005 IC50 = 5.67 nM T72841 CZ19RM 145949663 IC50 = 3810 nM T72841 CIKA61 145955698 IC50 = 4060 nM T72841 C8R6CB 145956201 IC50 = 610 nM T72841 C7Q8LS 145956663 IC50 = 3480 nM T72841 CX0K8G 145957185 IC50 = 45 nM T72841 CTOK38 145957219 IC50 = 3430 nM T72841 CI2V7N 145959169 IC50 = 3720 nM T72841 CIZE64 145960181 IC50 = 3040 nM T72841 CSB21A 145961412 IC50 = 4230 nM T72841 CZ56BE 149631187 IC50 = 4.33 nM T72841 C6QEZ8 150404085 IC50 = 20.33 nM T72841 C8U2LT 151011173 IC50 = 6 nM T72841 CJ54DK 151393167 IC50 = 4.67 nM T72841 CGY8C5 153534602 IC50 = 5.33 nM T72841 CA59FM 153534604 IC50 = 4.33 nM T72841 CV4FM2 153534607 IC50 = 7 nM T72841 C3M2NO 153534608 IC50 = 7.33 nM T72841 C7VS5G 155511937 IC50 > 10000 nM T72841 CVCK17 155513135 IC50 > 10000 nM T72841 C2PU1J 155513315 IC50 > 10000 nM T72841 CMQC26 155515404 IC50 > 10000 nM T72841 CP1L3J 155516697 IC50 > 10000 nM T72841 C36IUC 155517992 IC50 = 5.67 nM T72841 C82TWI 155524644 IC50 = 6.33 nM T72841 CO5YS6 155528287 IC50 = 11.33 nM T72841 CSLJ15 155528850 IC50 > 10000 nM T72841 CNZR30 155532489 IC50 = 5.33 nM T72841 C1YP5O 155533756 IC50 = 12.33 nM T72841 CC5HJ6 155535796 IC50 > 10000 nM T72841 CB3CY8 155538987 IC50 > 10000 nM T72841 CX63YO 155546410 IC50 = 7.67 nM T72841 CP72WM 155549027 IC50 = 9.33 nM T72841 CA5G2T 155551013 IC50 > 10000 nM T72841 C7AJZ5 155559268 IC50 > 10000 nM T72841 CPLW90 155561684 IC50 = 12.67 nM T72841 C9KY5I 155562382 IC50 = 8650 nM T72841 CWK95R 155565459 IC50 > 10000 nM T72841 CY71WP 155565677 IC50 > 10000 nM T72841 CMX67L 155567147 IC50 = 9700 nM T72841 D00QDE 135520118 IC50 = 3.6 nM T72841 D01TUB 135519319 IC50 = 4.6 nM T72841 D03CBX 135454802 IC50 = 4.3 nM T72841 D07XJC 135466462 IC50 = 46 nM T72841 D08SJL 135524856 IC50 = 75 nM T72841 D09FWS 135430317 IC50 = 52 nM T72841 D0E7RI 16122612 IC50 = 190 nM T72841 D0G3TK 5280863 IC50 = 9640 nM T72841 D0I1AF 135438472 IC50 = 22 nM T72841 D0K7HR 135409729 IC50 = 60 nM T72841 D0RD6G 135453199 IC50 = 52 nM T72841 D0W1YT 135466468 IC50 = 3.3 nM T72841 D0ZB7Z 6918788 IC50 = 270 nM T56272 CJKY76 7420 EC50 = 184000 nM T56272 CC2IU7 34037 EC50 > 1000000 nM T56272 CNXH01 231756 EC50 = 42000 nM T56272 CV6X3W 2734359 EC50 > 1000000 nM T56272 CY8JI4 2783146 EC50 > 1000000 nM T56272 CEFS70 7472024 EC50 > 1000000 nM T56272 CCK36A 11228924 EC50 = 38000 nM T56272 C9CK5H 13071646 EC50 = 16000 nM T56272 CE3W1R 15735511 EC50 = 129000 nM T56272 CIX0N5 19359201 EC50 > 1000000 nM T56272 C73XOY 21798667 EC50 > 1000000 nM T56272 CH7XV6 22052341 EC50 > 1000000 nM T56272 CZE7B8 53224766 EC50 > 1000000 nM T56272 C89RDH 66560365 EC50 > 1000000 nM T56272 CX5K1I 66560366 EC50 > 1000000 nM T56272 C4VB8Y 66560367 EC50 > 1000000 nM T56272 D0W1OR 7424 EC50 = 377000 nM T94085 D02DGU 444795 Ki = 0.1 nM T94085 D0BM5G 5381 EC50 = 63 nM T94085 D0G3PI 449171 EC50 = 21 nM T94085 D0JC9N 60164 EC50 = 22 nM T94085 D0N0RU 82146 EC50 = 6 nM T94085 D02GTY 108143 Ki = 6.5 nM T94085 D06FOU 11518241 EC50 = 500 nM T94085 D06QXI 9863342 EC50 > 1000 nM T94085 D0T3DO 9867758 EC50 = 200 nM T94085 D09YFJ 135411 Ki = 6500 nM T94085 D0M5EC 1714884 EC50 = 2511.89 nM T94085 D08GRF 5287705 Ki = 1.1 nM T94085 D0YO4D 3922 Ki = 1550 nM T94085 C7QAB1 2418 EC50 > 10000 nM T94085 CZBJ59 119342 Ki = 5.3 nM T94085 CWZY65 135754 Ki = 580 nM T94085 CRJ7K2 164456 Ki = 1120 nM T94085 C7AJR4 4433908 EC50 < 10000 nM T94085 CUL8F1 5354022 EC50 = 1000 nM T94085 C8ES5G 6366138 EC50 = 1100 nM T94085 C5EOB6 6366685 EC50 > 10000 nM T94085 CGL71X 6366726 EC50 > 0.001 nM T94085 C5EON6 6366727 EC50 > 0.001 nM T94085 C62YGF 6366732 EC50 > 0.001 nM T94085 CK4UA6 6366733 EC50 > 0.001 nM T94085 CLF4M5 6366734 EC50 = 2690 nM T94085 CA5GS8 6438168 EC50 > 0.001 nM T94085 C7C9SR 6439768 EC50 > 10000 nM T94085 CV6S9Y 6439770 EC50 = 11 nM T94085 C8WU1N 6440217 EC50 = 27 nM T94085 CG1S2D 6440346 EC50 = 24 nM T94085 C5LH2R 6441236 EC50 = 435 nM T94085 CJHW10 6441985 EC50 = 340 nM T94085 CHA3C2 6447986 EC50 = 1400 nM T94085 C3F4GD 6447987 EC50 = 740 nM T94085 CEV62Y 6450532 EC50 = 45 nM T94085 C31YCL 9797765 Ki = 6500 nM T94085 CBE62R 9799320 EC50 > 1000 nM T94085 CRK31P 9799442 EC50 > 10000 nM T94085 CENQ29 9799532 IC50 = 210 nM T94085 CSNI93 9799841 EC50 > 10000 nM T94085 CX2HY4 9801929 EC50 > 10000 nM T94085 CW7D0R 9810431 EC50 = 4 nM T94085 CUJ14W 9819890 EC50 > 10000 nM T94085 CEK1O4 9820039 EC50 = 210 nM T94085 CQI49S 9820393 EC50 > 10000 nM T94085 C7R9JM 9820462 Ki = 5787 nM T94085 C2X3PS 9822318 EC50 = 59 nM T94085 C6NGV0 9826896 IC50 = 4474 nM T94085 C94MFP 9842758 EC50 > 790 nM T94085 CI1P9A 9844563 Ki > 10000 nM T94085 CQFA96 9845057 Ki = 54 nM T94085 CE7D1J 9845382 IC50 = 6.5 nM T94085 CQ1ZH6 9847065 Ki = 2750 nM T94085 CA74MZ 9864886 IC50 = 220 nM T94085 C2ZY0W 9865875 EC50 = 112 nM T94085 CAE0R3 9868664 Ki = 4663 nM T94085 CRC51S 9869157 Ki = 6592 nM T94085 CA0TS6 9884959 EC50 = 733 nM T94085 CSK5B8 9885521 EC50 > 1000 nM T94085 CH0PV4 9885573 IC50 > 1000000 nM T94085 C3CS9R 9886082 EC50 > 10000 nM T94085 C5AD1H 9886137 Ki > 10000 nM T94085 CG3JR4 9887949 EC50 > 10000 nM T94085 C8V1ON 9888385 IC50 = 5.5 nM T94085 C90UXQ 9889347 Ki = 8300 nM T94085 C8MK1Y 9889522 Ki = 900 nM T94085 C2WFX1 9905729 Ki = 944 nM T94085 C2D9WJ 9906413 EC50 > 10000 nM T94085 C9AJZ7 9906514 EC50 = 59 nM T94085 C7E0IO 9907433 EC50 > 10000 nM T94085 CK9Z7I 9907650 IC50 = 2.2 nM T94085 CLP9A7 9909190 IC50 = 114 nM T94085 C0A3UZ 9911319 Ki = 4555 nM T94085 CSW2Y8 9929026 Ki > 1000 nM T94085 CQ6I7G 9946524 Ki > 1000 nM T94085 CIS1Z0 9948900 EC50 > 10000 nM T94085 C9VEF0 9949645 EC50 > 10000 nM T94085 C6CI3S 9950957 EC50 > 10000 nM T94085 CU46RB 9953712 Ki = 764 nM T94085 CL3BX4 9956886 EC50 = 290 nM T94085 C6JLI1 9973307 EC50 > 10000 nM T94085 C63OUJ 9976842 EC50 > 1000 nM T94085 CT7YJ8 9977495 EC50 = 94 nM T94085 C05EXS 9998870 EC50 > 10000 nM T94085 CL7X4Y 9999621 EC50 > 10000 nM T94085 CM1BQ5 10003577 Ki = 6756 nM T94085 CZP71W 10022432 IC50 = 100 nM T94085 CN6LP5 10022568 EC50 > 10000 nM T94085 C6L0XH 10044201 Ki = 487 nM T94085 CN0Y1P 10044591 EC50 = 8 nM T94085 CC4MF5 10045395 EC50 = 796 nM T94085 CE60FI 10065757 Ki > 1000 nM T94085 C2C0GJ 10066739 EC50 = 690 nM T94085 CVMD62 10069273 EC50 = 217 nM T94085 CFQ1Y3 10073992 Ki = 7280 nM T94085 C4VU6T 10087372 EC50 > 10000 nM T94085 CC8R9M 10093918 Ki = 980 nM T94085 C8MG7C 10094345 IC50 = 31.2 nM T94085 CSG68Q 10127015 IC50 = 20 nM T94085 CCKL65 10135144 Ki > 1000 nM T94085 CD3B1K 10135277 Ki > 1000 nM T94085 CQYW32 10137940 Ki = 6910 nM T94085 CU2H3N 10156587 Ki > 1000 nM T94085 C72HLB 10172878 IC50 = 83 nM T94085 C15HAE 10194688 IC50 = 20 nM T94085 C6KS9R 10202323 Ki = 8500 nM T94085 C9XS2G 10203771 Ki > 10000 nM T94085 CP96OH 10204841 Ki > 10000 nM T94085 CTKY45 10206438 Ki = 8360 nM T94085 C90YNI 10207221 Ki > 10000 nM T94085 C1O4PN 10207439 Ki > 10000 nM T94085 CZM6O3 10225147 Ki > 10000 nM T94085 CVL1Q6 10227224 Ki = 5000 nM T94085 C3IHN5 10251128 IC50 = 875 nM T94085 C1K8YO 10272875 Ki > 1000 nM T94085 CH5G4X 10273806 Ki = 6024 nM T94085 C0WRE7 10273807 Ki > 10000 nM T94085 CIKB68 10274731 Ki > 1000 nM T94085 CSE96Y 10292425 IC50 = 410000 nM T94085 C1LUP9 10294771 Ki > 10000 nM T94085 C27ZPC 10297135 Ki > 10000 nM T94085 CY1J5M 10308975 Ki > 1000 nM T94085 C9D7QC 10314719 EC50 = 0.6 nM T94085 C7G6XH 10315687 EC50 = 17 nM T94085 CVQ7Z6 10316839 EC50 > 10000 nM T94085 C6C5GP 10320109 Ki = 1600 nM T94085 C5LV9X 10358286 EC50 = 1000 nM T94085 CUEF37 10362997 IC50 > 1000 nM T94085 CG01ED 10383375 EC50 > 10000 nM T94085 CIK6T7 10384337 EC50 = 1128 nM T94085 CW39AL 10384413 IC50 = 225 nM T94085 CJCA73 10385620 Ki = 1144 nM T94085 C25HLM 10389354 Ki > 10000 nM T94085 CTO46Q 10405813 IC50 = 40 nM T94085 CXQ9S4 10450790 EC50 = 2856 nM T94085 CXA0N9 10458226 Ki = 1300 nM T94085 CV7C4F 10478196 IC50 = 1.5 nM T94085 C0KZT7 10519016 Ki = 834 nM T94085 CY62NU 10523459 Ki = 610 nM T94085 CQR8K0 10524574 IC50 = 2.4 nM T94085 C36OUF 10526963 Ki = 2000 nM T94085 CUO1I2 10543981 Ki = 130 nM T94085 C6CWZ1 10545954 EC50 = 620 nM T94085 C26NJB 10547547 IC50 = 19 nM T94085 C9EBZ0 10572606 IC50 = 130 nM T94085 CKBI92 10619546 IC50 = 32 nM T94085 CS96IV 10619935 EC50 = 14 nM T94085 C2HXP8 10641611 Ki = 1056 nM T94085 CMH87P 10643692 EC50 > 10000 nM T94085 CZ2C5K 10663499 Ki > 3000 nM T94085 C92TJP 10666483 Ki = 420 nM T94085 C1SNV6 10760998 Ki > 10000 nM T94085 C9UFH8 10763649 Ki = 460 nM T94085 C2TJY4 10788561 Ki > 10000 nM T94085 CTI5N7 10789247 Ki = 695 nM T94085 CMXI39 10804037 EC50 = 800 nM T94085 C8UG3F 10926235 EC50 > 500 nM T94085 CV38KY 11167904 EC50 > 10000 nM T94085 C34EXF 11221031 Ki = 93 nM T94085 CUP91B 11234875 Ki > 1000 nM T94085 C27ERO 11279584 IC50 = 20000 nM T94085 C8CS5F 11282651 IC50 > 30000 nM T94085 CT4HL6 11340230 IC50 = 470 nM T94085 CZ8IT7 11349121 IC50 = 100000 nM T94085 CF6XT3 11349910 Ki > 1000 nM T94085 CUY07B 11382535 IC50 > 1000000 nM T94085 C3FQ4D 11416475 EC50 = 57 nM T94085 CC5M6P 11416879 EC50 > 1000 nM T94085 CY6PJ9 11504066 EC50 = 103 nM T94085 CJH04T 11510627 EC50 = 270 nM T94085 CM34CL 11518525 EC50 = 180 nM T94085 C9NH8Y 11547131 EC50 = 1010 nM T94085 CQAF21 11554936 EC50 = 180 nM T94085 CLID54 11569584 EC50 > 10000 nM T94085 CZ4B9T 11612643 IC50 > 30000 nM T94085 CQ8S3K 11627002 EC50 = 200 nM T94085 C41AJB 11634244 EC50 > 10000 nM T94085 C3RMA0 11718697 EC50 > 10000 nM T94085 C0S9KJ 11740691 EC50 = 225 nM T94085 CY85CP 11749701 Ki > 1000 nM T94085 CFC0X5 11751490 IC50 < 1 nM T94085 C0WA5F 11793407 EC50 = 40 nM T94085 CD5K4U 11799011 Ki > 10000 nM T94085 CIZ52K 11948658 EC50 = 170 nM T94085 C7UWV3 12112296 EC50 = 989 nM T94085 CIQJ20 12112298 EC50 > 1000 nM T94085 CQ9YE5 12358678 EC50 = 102 nM T94085 C7JSH9 13833722 EC50 = 1100 nM T94085 C7Z0YT 13833727 EC50 = 2300 nM T94085 CY2OL5 14259057 EC50 = 1700 nM T94085 CN7CX1 14726558 IC50 = 0.45 nM T94085 C8DP6M 14776682 EC50 = 420 nM T94085 CQI17S 15160092 EC50 = 240 nM T94085 CNS9T8 15434197 Ki > 1000 nM T94085 CDA7J9 15951925 EC50 < 10000 nM T94085 C4LRI8 15951927 EC50 < 10000 nM T94085 C9S5XT 15952013 EC50 < 10000 nM T94085 C5J3ZE 16661643 EC50 = 40 nM T94085 CX6L0G 16661644 EC50 = 43 nM T94085 C5GTA2 18507967 EC50 = 2300 nM T94085 CQYD01 18768139 EC50 = 212 nM T94085 CX3Q7D 20243100 EC50 = 15 nM T94085 C5MHX3 21217837 Ki = 821 nM T94085 CV1C4A 22226112 EC50 > 1000 nM T94085 CTE1N2 24748569 EC50 > 10000 nM T94085 CSTR97 25259041 EC50 = 1995.26 nM T94085 CT2B1Z 25259265 EC50 = 1584.89 nM T94085 C2G6QF 25259266 EC50 = 15.1 nM T94085 CS7U6L 44285287 EC50 = 550 nM T94085 CPA87R 44287651 Ki > 10000 nM T94085 C1K8FB 44287715 Ki > 10000 nM T94085 CI83JY 44287875 Ki = 1786 nM T94085 CB8PI2 44304045 Ki > 1000 nM T94085 CFTB98 44313143 Ki = 1471 nM T94085 C4E1OW 44313513 Ki > 3000 nM T94085 C8W6JP 44314319 Ki = 3.1 nM T94085 C17LMT 44314320 Ki > 4000 nM T94085 C92VTZ 44316277 EC50 = 2300 nM T94085 CIVH74 44316525 Ki > 1000 nM T94085 CAP68W 44316543 Ki > 1000 nM T94085 CAI2Z5 44316544 Ki > 1000 nM T94085 C0YQ8H 44316756 Ki > 1000 nM T94085 C6Q1CA 44316796 Ki > 1000 nM T94085 CLK5H0 44316811 Ki > 1000 nM T94085 CXV0B4 44321951 EC50 = 2100 nM T94085 C1KUN0 44325759 Ki > 1000 nM T94085 CLB6X7 44325767 Ki > 1000 nM T94085 CW0T6K 44353336 Ki = 4555 nM T94085 C8K0AB 44353347 Ki = 3730 nM T94085 C3DYE9 44353422 Ki > 10000 nM T94085 C5DTY3 44353441 Ki > 10000 nM T94085 C2M8TN 44353456 Ki > 10000 nM T94085 CVKA40 44353466 Ki = 4659 nM T94085 C8J5SA 44353480 Ki = 2500 nM T94085 CIB15X 44353481 Ki > 10000 nM T94085 C3MY4C 44364348 Ki = 8500 nM T94085 CY9XP2 44366042 EC50 > 10000 nM T94085 CT3S5O 44377822 EC50 = 30 nM T94085 C5QRI4 44401302 IC50 = 11.1 nM T94085 CJVG73 44459626 EC50 = 5000 nM T94085 CR5SI0 44476535 EC50 > 10000 nM T94085 CP4DM5 44581289 EC50 > 1000 nM T94085 C8UHG5 45270032 IC50 = 15 nM T94085 CN9L7G 46916268 EC50 > 8300 nM T94085 CUD91T 49862248 EC50 > 10000 nM T94085 C9G4IT 60729785 EC50 = 77.5 nM T94085 CZ38NM 69588033 EC50 = 34 nM T94085 CN03UB 71568951 EC50 = 82 nM T94085 CX9EA0 71568952 EC50 = 88.9 nM T94085 C4GRK9 71571262 EC50 = 8.2 nM T94085 CVW1H0 73350281 Ki > 10000 nM T94085 C9W0ZA 86276176 EC50 = 110 nM T94085 CBN9F0 101616167 EC50 = 65 nM T94085 C6TBD2 121345502 EC50 > 20000 nM T94085 C6L4GM 135949402 EC50 > 1000 nM T94085 C5L6AU 136126668 EC50 > 1000 nM T94085 CN5MO3 136126669 EC50 > 1000 nM T94085 CJ5EH7 136126670 EC50 > 1000 nM T94085 CI4CG1 136126671 EC50 = 520 nM T94085 CAF61N 136249387 IC50 = 1277 nM T94085 CB32UM 136264284 IC50 = 2650 nM T94085 C1J4DV 145965542 EC50 = 11 nM T94085 CRKW68 145966900 EC50 > 10000 nM T94085 C4MY5N 145967331 EC50 = 336 nM T94085 CC05VW 145970742 EC50 > 10000 nM T94085 CDBR75 145976745 EC50 = 317 nM T94085 C2A1UC 10429766 Ki > 1000 nM T94085 D09RRF 11530459 EC50 = 630.96 nM T94085 D0F8CC 10090192 EC50 = 370 nM T94085 D0F8JO 9951075 IC50 = 20000 nM T94085 D0G6JM 5289501 EC50 = 0.18 nM T94085 D0P0PP 10044792 IC50 = 10 nM T94085 D0Q0IR 177238 IC50 = 31 nM T94085 D0Q9FZ 6442223 EC50 = 4 nM T94085 D0RD0R 2126 EC50 = 0.3 nM T94085 D0X5WP 10410894 Ki = 1400 nM T72252 D01YIF 135421197 EC50 = 4500 nM T72252 D0J3SU 9847835 Ki = 6 nM T72252 CY0FV4 17520 IC50 = 137400 nM T72252 COW5R3 608841 Ki = 6200 nM T72252 C5WKA9 2779120 IC50 = 46000 nM T72252 C1V6CM 2821593 IC50 = 170000 nM T72252 C7CLA9 2821595 IC50 > 200000 nM T72252 C2U4HS 2821632 IC50 > 200000 nM T72252 CMP1F6 2821634 IC50 > 200000 nM T72252 CR7N4T 2821636 IC50 > 200000 nM T72252 COTB47 2821639 IC50 > 200000 nM T72252 C1JRB7 2821640 IC50 > 200000 nM T72252 C12EXP 2821660 IC50 > 200000 nM T72252 CGOH73 2821679 IC50 > 200000 nM T72252 C1RUH9 4246483 IC50 = 84900 nM T72252 CT4YC1 5287959 IC50 = 24 nM T72252 C3T8NF 5288850 Ki = 47 nM T72252 CO58XD 5311161 IC50 > 100000 nM T72252 C1KR5B 5327301 Ki = 190 nM T72252 C37TKL 5327302 Ki = 470 nM T72252 C64ZMN 5327304 Ki = 130 nM T72252 C3IZ2W 5327307 Ki = 90 nM T72252 C16DTL 5327308 Ki = 120 nM T72252 C4O3QY 5327309 Ki = 130 nM T72252 C3GUM7 5327310 Ki = 940 nM T72252 C3LZX9 8027611 IC50 > 20000 nM T72252 CFN2P6 9800285 Ki = 47 nM T72252 CE7I9W 9806986 IC50 = 1.13 nM T72252 CYFG94 9807028 IC50 = 3200 nM T72252 CD3P2F 9807170 IC50 = 0.75 nM T72252 C3S1EP 9807375 IC50 > 10 nM T72252 C13PRZ 9809421 IC50 = 120 nM T72252 CLTO67 9821317 IC50 = 7 nM T72252 C4XO3K 9821545 Ki = 47 nM T72252 C6S3KT 9840223 IC50 = 170 nM T72252 CN02PU 9849845 IC50 = 4.68 nM T72252 C5MCX4 9849846 IC50 > 10 nM T72252 CDC86G 9850642 IC50 > 10 nM T72252 CJO3A5 9851213 IC50 = 2.42 nM T72252 C56LDH 9851279 IC50 = 97 nM T72252 C6O0QH 9852052 IC50 = 0.008 nM T72252 C2N3LE 9871540 IC50 > 10 nM T72252 CX17DM 9871570 IC50 = 9.71 nM T72252 CF0V7B 9871631 IC50 = 0.49 nM T72252 CLQH78 9892350 IC50 = 9.73 nM T72252 CW75OE 9892652 IC50 = 5.17 nM T72252 C3YAL4 9895375 IC50 = 8.4 nM T72252 C2DMG1 9914167 IC50 = 21.8 nM T72252 CK15RJ 9916276 IC50 = 3.28 nM T72252 C0D2IJ 9936767 IC50 = 0.81 nM T72252 CG90WC 9939287 IC50 = 360 nM T72252 CFCK64 9939773 IC50 = 2300 nM T72252 CN63JG 9958554 IC50 = 2.54 nM T72252 C9CV0Y 10001828 IC50 = 1810 nM T72252 CW4Q3N 10031194 IC50 = 2500 nM T72252 CHWA42 10074552 IC50 = 1800 nM T72252 CZ3IH4 10414828 IC50 > 10000 nM T72252 CX67SZ 10826725 Ki = 170 nM T72252 CDX7A4 10963183 Ki = 90 nM T72252 C2GPV7 11150874 IC50 = 30.87 nM T72252 C6EL1S 11197291 IC50 = 1050 nM T72252 CM8O6L 11257152 IC50 = 11 nM T72252 CCV6T0 11374367 IC50 = 10 nM T72252 C4F8DC 11444079 IC50 = 1.8 nM T72252 CDT9G3 11467504 IC50 = 0.09 nM T72252 CV4CP9 11496333 IC50 = 29.5 nM T72252 CGE2J0 11497112 IC50 = 26.7 nM T72252 C6IS9K 11509289 IC50 = 362.5 nM T72252 C6L2MY 11509300 IC50 = 214.9 nM T72252 CC31QO 11509301 IC50 = 142.3 nM T72252 CS8OX7 11510566 IC50 = 4 nM T72252 C7FY9B 11512139 IC50 = 34.8 nM T72252 C15VFG 11515586 IC50 = 304 nM T72252 CW6PC0 11519268 IC50 = 41 nM T72252 CZC5D9 11525874 IC50 = 22.7 nM T72252 C5BNE1 11533326 IC50 = 14.5 nM T72252 CDK3Z5 11533935 IC50 = 5.9 nM T72252 C4IC7E 11541867 IC50 = 13.8 nM T72252 C3USR9 11543714 IC50 = 139 nM T72252 C3P2GZ 11548424 IC50 = 69.8 nM T72252 CVX4M6 11548909 IC50 = 18.6 nM T72252 C17OJS 11572844 IC50 = 136 nM T72252 CF0V3P 11576540 IC50 = 14.1 nM T72252 C1T9DY 11576622 IC50 = 135 nM T72252 C03KPR 11576852 EC50 = 19.8 nM T72252 CN67DR 11583840 IC50 = 21 nM T72252 CPD0M8 11584106 IC50 = 58 nM T72252 CL16IM 11591540 IC50 = 15.1 nM T72252 CE2TX6 11591919 IC50 = 25.7 nM T72252 CG4Z9A 11598106 IC50 = 4.6 nM T72252 CV6MF1 11614728 IC50 = 42.8 nM T72252 CFP19E 11619968 IC50 = 17 nM T72252 CA0LH6 11624920 IC50 = 1350 nM T72252 CEY39D 11628992 IC50 = 50.9 nM T72252 C6UAV3 11632008 IC50 = 63 nM T72252 C6Y5MG 11634372 IC50 = 26 nM T72252 CKJE92 11634649 IC50 = 22.2 nM T72252 C91JNO 11639020 IC50 = 64 nM T72252 C4MCW2 11646889 IC50 = 218 nM T72252 C2KFU3 11647018 IC50 = 94.9 nM T72252 CH20JE 11652994 IC50 = 2710 nM T72252 CN32TX 11664423 IC50 = 366 nM T72252 CUD05C 11670894 IC50 = 23.3 nM T72252 CX97NT 11684618 IC50 = 23.2 nM T72252 C05YRV 11699954 IC50 = 42 nM T72252 CKEX64 11700402 IC50 = 29.2 nM T72252 C89COT 11705942 IC50 = 15.1 nM T72252 C86PAH 11712912 IC50 = 44 nM T72252 C7QK5F 11755713 IC50 = 2700 nM T72252 C7YI1R 16725993 IC50 = 8 nM T72252 CXH9M5 16749067 IC50 = 1585 nM T72252 C2DJ5W 16749068 IC50 = 11.7 nM T72252 COM07G 16749069 IC50 = 785 nM T72252 CPG8Q0 16749161 IC50 = 126 nM T72252 CG84TK 16749162 IC50 = 32.8 nM T72252 CT3HD1 16749163 IC50 = 28.3 nM T72252 CZM4X2 16749164 IC50 = 29.6 nM T72252 CUZ8N4 16749267 IC50 = 34.8 nM T72252 CMEK96 16749268 IC50 = 6.6 nM T72252 C01HBN 16749269 IC50 = 51.7 nM T72252 CWG3C8 16749270 IC50 = 92.2 nM T72252 C8R3GD 16749271 IC50 = 26.3 nM T72252 CW9HL5 23645230 IC50 = 3100 nM T72252 C5G2IL 23645238 IC50 = 3625 nM T72252 C74OPE 23645239 IC50 = 8360 nM T72252 CK7B2A 23645240 IC50 = 1050 nM T72252 C8YA0T 23645241 IC50 = 10860 nM T72252 C8J7UY 23645242 IC50 > 10000 nM T72252 C3MGC1 23645243 IC50 = 3405 nM T72252 CLSU45 23645244 IC50 > 10000 nM T72252 C95KHP 23645245 IC50 = 2760 nM T72252 C08UYG 23645246 IC50 > 10000 nM T72252 C6YEO7 23645247 IC50 > 10000 nM T72252 CFH23D 23645248 IC50 = 10860 nM T72252 CY0M3Z 23645249 IC50 = 5095 nM T72252 C4TIM0 23645250 IC50 > 10000 nM T72252 CZ9HT6 23645253 IC50 = 130 nM T72252 CZ59CM 23645306 IC50 = 1500 nM T72252 CNU1R6 23645307 IC50 = 1400 nM T72252 C8WF2G 23645308 IC50 = 3100 nM T72252 CBSA54 23645309 IC50 = 1700 nM T72252 CTI80F 25178948 EC50 = 13.5 nM T72252 C2GI4J 25178949 EC50 = 16.8 nM T72252 CQ2GM9 25178950 EC50 = 14.4 nM T72252 C4GFV6 25179140 EC50 = 60.4 nM T72252 CYL36B 25179141 EC50 = 2.2 nM T72252 CGC69Q 25179143 EC50 = 78.6 nM T72252 C27YJF 25179144 EC50 = 28.2 nM T72252 C2YTB7 25179145 EC50 = 18.3 nM T72252 C6GTV3 25179324 EC50 = 8 nM T72252 CIC46T 25179513 EC50 = 13 nM T72252 CK96WB 25179514 EC50 = 2.3 nM T72252 CGX78D 25217029 IC50 = 50 nM T72252 CW2L9Q 25217030 IC50 = 26.5 nM T72252 C8UTC4 25217031 IC50 = 45 nM T72252 CZ43KQ 25217032 IC50 = 96.3 nM T72252 C2P9NI 25217145 IC50 = 26.1 nM T72252 C8C9XU 42618276 IC50 = 2233 nM T72252 CFO93N 42618277 IC50 = 1483 nM T72252 CS1KQ0 42618278 IC50 = 878 nM T72252 CVI16X 42618279 IC50 = 1147 nM T72252 C3MRA0 42618280 IC50 = 3416 nM T72252 C8UO9S 42618281 IC50 = 4467 nM T72252 C68NPR 42618282 IC50 = 4100 nM T72252 CL41SD 42618283 IC50 = 7900 nM T72252 CJ7U2E 42618284 IC50 = 1625 nM T72252 CZL8C7 42618285 IC50 = 1893 nM T72252 CNIQ28 42618286 IC50 = 5100 nM T72252 C91OMB 42618287 IC50 = 132 nM T72252 C5AC1L 42618288 IC50 = 248 nM T72252 CFU5T2 42618289 IC50 = 471 nM T72252 CK9H3M 42618290 IC50 = 340 nM T72252 CV4H2J 42618291 IC50 = 587 nM T72252 C7VPU3 42618292 IC50 = 443 nM T72252 C6R2FM 42618293 IC50 = 471 nM T72252 C4QOV7 44157030 IC50 = 58 nM T72252 CGB3E4 44157031 IC50 = 8.1 nM T72252 CT2B8Z 44157032 IC50 = 6.8 nM T72252 CT7VO2 44157085 IC50 = 68 nM T72252 CWMU91 44157086 IC50 = 99 nM T72252 C6LZ5Y 44157087 IC50 = 61 nM T72252 CYSJ79 44157089 IC50 = 1.9 nM T72252 CMX7W1 44157090 IC50 = 2.4 nM T72252 C35DAU 44158016 IC50 = 1660 nM T72252 C7B3VE 44158086 IC50 = 16 nM T72252 C20WEJ 44158089 IC50 = 349 nM T72252 C68KOD 44158154 IC50 = 7.6 nM T72252 C4C1RU 44158155 IC50 = 5 nM T72252 CN1YR9 44158157 IC50 = 43 nM T72252 C80XPD 44158237 IC50 = 61 nM T72252 CN09UV 44158238 IC50 = 24 nM T72252 CT9DF4 44158240 IC50 = 50 nM T72252 CHDF62 44158242 IC50 = 111 nM T72252 CS6X1C 44158325 IC50 = 7.2 nM T72252 C17TEZ 44158326 IC50 = 0.6 nM T72252 CZ0VT3 44158328 IC50 = 9 nM T72252 CD8WB9 44304162 Ki = 10000 nM T72252 CAB39E 44331552 IC50 = 4160 nM T72252 CE0FW4 44331565 IC50 = 3610 nM T72252 C8SZN9 44331566 IC50 = 3380 nM T72252 CMFW61 44331567 IC50 = 4080 nM T72252 CHYL38 44331577 IC50 = 5890 nM T72252 C1I9QH 44331578 IC50 = 4410 nM T72252 C4VGZ1 44331579 IC50 = 3360 nM T72252 CRZ01H 44331580 IC50 = 12000 nM T72252 CFOR90 44331674 IC50 = 3750 nM T72252 CK7VI8 44331675 IC50 = 2020 nM T72252 CH7GS4 44331676 IC50 > 10000 nM T72252 C4FOD3 44331693 IC50 = 6040 nM T72252 CJY5L2 44331739 IC50 = 2310 nM T72252 C8N2GQ 44331740 IC50 = 2740 nM T72252 CW9K4Q 44331815 IC50 = 1490 nM T72252 CT76DG 44331816 IC50 = 7250 nM T72252 CC70GF 44331830 IC50 = 680 nM T72252 CNJ19L 44331876 IC50 > 10000 nM T72252 C46IPA 44331879 IC50 > 10000 nM T72252 CP0Y8M 44331898 IC50 = 10 nM T72252 CF3R6W 44331908 IC50 > 10000 nM T72252 C0S8LV 44331910 IC50 = 10 nM T72252 CTM5W1 44331914 IC50 = 130 nM T72252 C0YZ9O 44331915 IC50 = 587 nM T72252 CPZ7Q2 44331933 IC50 = 7270 nM T72252 C4NK1S 44331942 IC50 = 10 nM T72252 CXKY19 44331943 IC50 = 8870 nM T72252 C3FC8D 44331944 IC50 > 10000 nM T72252 CH1ZF2 44331953 IC50 = 2920 nM T72252 C0QJ8V 44331957 IC50 = 37030 nM T72252 C1HBX6 44331963 IC50 = 21900 nM T72252 C7UXK5 44331964 IC50 = 6810 nM T72252 C42PGN 44331965 IC50 = 2670 nM T72252 C5J7KX 44331966 IC50 > 10000 nM T72252 CG83FS 44331967 IC50 = 1510 nM T72252 CGAJ95 44331977 IC50 = 10900 nM T72252 CCYX84 44331980 IC50 = 2100 nM T72252 C5UIO2 44331987 IC50 = 8240 nM T72252 C0PM5C 44332004 IC50 = 8770 nM T72252 C4ENB1 44332005 IC50 = 11000 nM T72252 CFK4Z1 44332024 IC50 = 1320 nM T72252 CTM3G2 44332026 IC50 = 3600 nM T72252 C48ZEW 44332028 IC50 = 4570 nM T72252 C30MKG 44332029 IC50 = 34700 nM T72252 C7OS9X 44332050 IC50 = 2200 nM T72252 C9Y6NP 44332051 IC50 = 9720 nM T72252 C0VGF8 44332058 IC50 = 2790 nM T72252 CQU84D 44332068 IC50 = 6820 nM T72252 CBL91D 44332078 IC50 = 5230 nM T72252 C4VCM3 44332093 IC50 = 9650 nM T72252 C92QVT 44332108 IC50 = 1740 nM T72252 CQLZ09 44332109 IC50 = 32400 nM T72252 C4CUL6 44332112 IC50 = 43660 nM T72252 CN2YM6 44332113 IC50 = 17000 nM T72252 C4CY8K 44332118 IC50 = 6140 nM T72252 CXZ2N1 44332120 IC50 = 3480 nM T72252 CD56PK 44332121 IC50 = 3850 nM T72252 C5A6OJ 44332128 IC50 = 18200 nM T72252 C6IZ2R 44332129 IC50 = 2520 nM T72252 C5DY0G 44332136 IC50 = 1650 nM T72252 CQ1K9H 44332311 IC50 = 1320 nM T72252 C9LOS2 44332330 IC50 = 1370 nM T72252 C2U6GB 44332331 IC50 = 7430 nM T72252 CH01QW 44332332 IC50 = 11300 nM T72252 C8D5TB 44364680 Ki = 90 nM T72252 CV23MO 44389236 IC50 = 0.54 nM T72252 C2I3VJ 44389240 IC50 = 0.01 nM T72252 CI89LR 44389245 IC50 = 0.31 nM T72252 CR7VM8 44389295 IC50 > 10 nM T72252 CU5VW3 44389297 IC50 = 1.04 nM T72252 C5P8TU 44389299 IC50 = 1.01 nM T72252 C5YC0O 44389306 IC50 = 0.41 nM T72252 C1FMX8 44389307 IC50 = 3.24 nM T72252 CB6US3 44389310 IC50 = 2.6 nM T72252 CC8S0I 44389315 IC50 = 0.73 nM T72252 CEO19T 44389316 IC50 = 0.54 nM T72252 CRC82Z 44389318 IC50 > 10 nM T72252 CPE0S2 44389319 IC50 = 0.13 nM T72252 CC8MG3 44389324 IC50 = 0.12 nM T72252 C9X1RJ 44389325 IC50 = 1 nM T72252 CF0CN3 44389326 IC50 = 0.32 nM T72252 C7LQP0 44389331 IC50 = 0.26 nM T72252 CEQ2L1 44389335 IC50 > 10 nM T72252 C9C3JB 44389337 IC50 = 0.13 nM T72252 CU0I3N 44389338 IC50 = 0.083 nM T72252 CALT41 44389340 IC50 = 0.48 nM T72252 C5LO3T 44389347 IC50 = 0.13 nM T72252 CJA5K7 44389348 IC50 = 0.84 nM T72252 C2WS9G 44389351 IC50 = 0.14 nM T72252 CEH8Z5 44389369 IC50 = 0.14 nM T72252 CBJ15U 44389458 IC50 = 0.11 nM T72252 C2OU7Z 44389483 IC50 = 0.1 nM T72252 CA81WI 44389513 IC50 = 0.6 nM T72252 CL4G2Y 44389531 IC50 = 0.065 nM T72252 CX5Y3A 44389532 IC50 = 0.042 nM T72252 CEH02Q 44389544 IC50 = 0.087 nM T72252 CXN03I 44389545 IC50 = 0.036 nM T72252 CQPY50 44391346 IC50 = 2215 nM T72252 CJQE23 44391364 IC50 = 3690 nM T72252 CE3YN5 44391369 IC50 > 10000 nM T72252 CWVF04 44391384 IC50 = 5300 nM T72252 C0J6SU 44391388 IC50 = 4200 nM T72252 C24KOF 44391455 IC50 = 10000 nM T72252 CA58XR 44391530 IC50 = 545 nM T72252 CU3ZB5 44391569 IC50 = 91 nM T72252 CI7F3G 44391602 IC50 = 290 nM T72252 CL73OE 44391603 IC50 = 63 nM T72252 CIU0P1 44391632 IC50 = 135 nM T72252 CJ6QG4 44417479 IC50 = 32.3 nM T72252 C7RX9I 44418960 Ki = 1200 nM T72252 CXR1V5 44434249 IC50 = 11 nM T72252 C31JIN 44438441 IC50 = 3490 nM T72252 CKI30F 44438442 IC50 = 920 nM T72252 CNO1C0 44438443 IC50 = 800 nM T72252 CI1G7O 44438444 IC50 = 280 nM T72252 C9SN7W 44572193 IC50 > 100000 nM T72252 C17DXL 44572194 IC50 > 100000 nM T72252 CMJN04 44572195 IC50 = 123 nM T72252 CV69UW 44572196 IC50 = 40 nM T72252 C2MY8P 44572210 IC50 = 100 nM T72252 CUD5Q6 44572270 IC50 = 111 nM T72252 C4K3YQ 44572673 IC50 = 319 nM T72252 C3LYN7 44572674 IC50 = 79 nM T72252 CK4P3D 44572710 IC50 = 52 nM T72252 C62IOT 44572711 IC50 = 217 nM T72252 CZMC41 44572712 IC50 = 129 nM T72252 CZ6Y1F 44572713 IC50 = 11 nM T72252 CL5E3R 44572714 IC50 = 29 nM T72252 C1TD7H 44572774 IC50 = 2940 nM T72252 CJQ0M7 44572775 IC50 = 1440 nM T72252 CRY8Z1 44572776 IC50 = 28 nM T72252 C9YZ1J 44572777 IC50 = 266 nM T72252 C4PZ2Q 44572967 IC50 = 178 nM T72252 CH6N1M 44572968 IC50 = 44 nM T72252 CI71AG 44572969 IC50 = 11 nM T72252 CNR7O3 44572970 IC50 = 135 nM T72252 C1IZ3B 44573088 IC50 > 100000 nM T72252 CRK8D6 44573089 IC50 = 5640 nM T72252 CA4TE6 44573090 IC50 = 113000 nM T72252 CA7QH2 44573091 IC50 = 19400 nM T72252 CV34ZB 46933021 IC50 > 200000 nM T72252 C3HRL2 46933163 IC50 > 200000 nM T72252 CL4I1F 46933460 IC50 > 200000 nM T72252 CM5T3U 46933463 IC50 > 200000 nM T72252 C7JW2B 46933464 IC50 > 200000 nM T72252 C82LPS 46933615 IC50 > 200000 nM T72252 CDY2W5 49796910 IC50 = 0.013 nM T72252 C0HMT1 49797331 IC50 = 64.7 nM T72252 C3M2BW 52918163 IC50 = 17.6 nM T72252 CF24IM 52918177 IC50 = 11.3 nM T72252 CR9I7F 52918178 IC50 = 3.8 nM T72252 C2VPU1 52918179 IC50 = 6.1 nM T72252 C47TKY 52948065 IC50 > 200000 nM T72252 C8Z2TQ 54580470 IC50 = 28.9 nM T72252 CMU0B4 54581481 IC50 = 11.9 nM T72252 CCS8Y3 54581987 IC50 = 70 nM T72252 CJEP38 54582484 IC50 = 17.6 nM T72252 C61NWL 54582924 IC50 = 12.3 nM T72252 CO0AG3 54583923 IC50 = 292 nM T72252 CI2DL4 54583924 IC50 = 15.4 nM T72252 CV2WU1 54583925 IC50 = 15.3 nM T72252 CXA51D 54584867 IC50 = 18 nM T72252 C8YSL0 54585834 IC50 = 68.3 nM T72252 C9B5OF 54586343 IC50 = 19.2 nM T72252 C7A8ER 54587376 IC50 = 10.2 nM T72252 CGY3W2 71471109 IC50 = 150 nM T72252 CKZ2H0 71582971 IC50 = 540 nM T72252 C4WJ5F 71582972 IC50 = 24.6 nM T72252 CXA62J 71582973 IC50 = 12.3 nM T72252 CNZS31 71582974 IC50 = 125 nM T72252 CE4L9D 71582975 IC50 = 515 nM T72252 CXMS80 71583078 IC50 = 33.7 nM T72252 C30UIL 71583079 IC50 = 13.2 nM T72252 CJBC14 71583080 IC50 = 64.6 nM T72252 C57MOP 71583081 IC50 = 218 nM T72252 CS0YK9 71583082 IC50 = 1330 nM T72252 C3UTO9 71583083 IC50 = 39.6 nM T72252 CW1R5Q 71583084 IC50 = 9.68 nM T72252 CR57LS 71583192 IC50 = 1420 nM T72252 C8B3NZ 71583193 IC50 = 7.47 nM T72252 CB6DY7 71583194 IC50 = 265 nM T72252 C7Q2ZN 71682003 IC50 = 128 nM T72252 CV96GT 71682004 IC50 = 103 nM T72252 C82YPX 71682161 IC50 = 296 nM T72252 CM76CD 71682162 IC50 = 27 nM T72252 CY07ID 71682310 IC50 = 71 nM T72252 CZI7D3 71682311 IC50 = 0.951 nM T72252 CJLY24 71698534 IC50 = 14900 nM T72252 CP3GS5 71698535 IC50 = 178 nM T72252 C6E5OV 71698716 IC50 > 500000 nM T72252 C9V4WS 71698717 IC50 > 500000 nM T72252 C26LVZ 71698718 IC50 > 500000 nM T72252 CAJ2N7 71698719 IC50 > 500000 nM T72252 C4CYG0 71698720 IC50 = 26400 nM T72252 C0ANH2 71698798 IC50 > 500000 nM T72252 C9O0CY 71698799 IC50 = 59600 nM T72252 C7CUJ8 71698800 IC50 = 42600 nM T72252 CIW75R 71698803 IC50 > 500000 nM T72252 CUM83A 71698883 IC50 = 52700 nM T72252 C2S7VN 71698884 IC50 = 78300 nM T72252 CP4Y9M 71698885 IC50 = 67700 nM T72252 CR4O3U 71698886 IC50 = 147000 nM T72252 CWDZ96 71698887 IC50 = 8460 nM T72252 CFP6Y2 71698973 IC50 = 12100 nM T72252 CIG39A 71698974 IC50 = 1880 nM T72252 C25YSR 71698975 IC50 = 1250 nM T72252 CG04WQ 71698976 IC50 > 500000 nM T72252 CR24DS 71698977 IC50 = 11900 nM T72252 C6PO1L 71698978 IC50 > 500000 nM T72252 CX1GO2 71699066 IC50 = 47800 nM T72252 CANH70 71716242 IC50 = 500 nM T72252 C40WIR 71718085 IC50 = 23700 nM T72252 CU75VK 71719897 IC50 > 100000 nM T72252 CBV6F1 71720507 IC50 = 24500 nM T72252 CGL6T9 73347421 IC50 > 500000 nM T72252 CBF89G 73353489 IC50 > 500000 nM T72252 CKYI28 73354985 IC50 > 500000 nM T72252 C4U5TO 76311196 IC50 = 16.5 nM T72252 CSI53E 76311200 IC50 = 14.2 nM T72252 CNOL37 76311201 IC50 = 24 nM T72252 C8IS5Q 76314800 IC50 = 19.8 nM T72252 CK41QI 76314804 IC50 = 21.8 nM T72252 CHS61N 76314805 IC50 = 9.6 nM T72252 CDY7K0 76318413 IC50 = 5.4 nM T72252 CB2N6G 76322078 IC50 = 3512 nM T72252 C8SPW6 76322082 IC50 = 14 nM T72252 CC2EP6 76325698 IC50 = 15.9 nM T72252 CFY79U 76332916 IC50 = 11.2 nM T72252 CD35SI 76332917 IC50 = 25.3 nM T72252 C3FQX0 76336535 IC50 = 41.4 nM T72252 CV4PE6 76336536 IC50 = 20.4 nM T72252 CQ46DF 86279277 IC50 = 164 nM T72252 C0FDU4 86279278 IC50 = 248000 nM T72252 C75MZK 90654525 IC50 = 418.7 nM T72252 CL2E7D 90654526 IC50 = 390.2 nM T72252 CMN74D 90654527 IC50 = 9.424 nM T72252 C2CUV9 90654528 IC50 = 637.9 nM T72252 C3OC8I 90654529 IC50 = 75.82 nM T72252 C21PEL 90654530 IC50 = 64.44 nM T72252 CTFA68 90654531 IC50 = 72.2 nM T72252 CY63ON 90654532 IC50 = 156.1 nM T72252 CY8HP0 90654533 IC50 = 156.7 nM T72252 CHO1G0 90654534 IC50 = 4794 nM T72252 COR17A 90654535 IC50 = 193.9 nM T72252 CLB31J 90654536 IC50 = 100400 nM T72252 C5Y6OL 90654537 IC50 = 2590 nM T72252 CP45YW 90654538 IC50 = 1350 nM T72252 CB0YI1 90654539 IC50 = 6070 nM T72252 C4YKM7 90654540 IC50 = 94.98 nM T72252 CKCI60 90663142 IC50 = 7240 nM T72252 C43QKY 101879103 IC50 = 54 nM T72252 CW02EX 101879104 IC50 = 51.9 nM T72252 C3SUH2 118723310 IC50 = 500000 nM T72252 C3M5TO 118723311 IC50 = 10500 nM T72252 CX82RL 118723312 IC50 = 20.1 nM T72252 C0SIK1 118723313 IC50 = 42.4 nM T72252 C3GPO7 118723314 IC50 = 907 nM T72252 C8H0EL 118723315 IC50 = 123 nM T72252 CTE1O2 118723316 IC50 = 68.1 nM T72252 CE8O9P 118723317 IC50 = 279 nM T72252 C3UZ6B 118723318 IC50 = 500000 nM T72252 C15RJF 118723319 IC50 = 553 nM T72252 C0OIE9 118723320 IC50 = 135 nM T72252 C01SDY 118723321 IC50 = 157 nM T72252 C0X9MJ 118723322 IC50 = 3.3 nM T72252 C5LB3W 118723323 IC50 = 20.1 nM T72252 C1GQO9 118723324 IC50 = 5.95 nM T72252 C48DEF 118723325 IC50 = 22.7 nM T72252 C67QMY 118723326 IC50 = 500000 nM T72252 CCJ27M 118723327 IC50 = 263 nM T72252 COG92V 118723328 IC50 = 55.7 nM T72252 CSX85P 118723329 IC50 = 6620 nM T72252 CICB42 118723330 IC50 = 9.7 nM T72252 C13BRQ 118723331 IC50 = 39.3 nM T72252 CDM0A7 118724007 IC50 = 268.7 nM T72252 CE01XH 118724008 IC50 = 370.3 nM T72252 C3MCW6 118724009 IC50 = 184 nM T72252 C9X0ZM 118724010 IC50 = 182.3 nM T72252 CNA7D6 118724011 IC50 = 207.2 nM T72252 CBWT97 118724012 IC50 = 211.2 nM T72252 CQA8U6 118724013 IC50 = 213.3 nM T72252 C12EHA 118724014 IC50 = 123 nM T72252 CNB6M9 118724015 IC50 = 457.7 nM T72252 CL9AS6 118724016 IC50 = 608.1 nM T72252 CX9D0V 118724017 IC50 = 144.9 nM T72252 CXT5V4 118724018 IC50 = 607.1 nM T72252 C6Q1IG 118724019 IC50 = 585.6 nM T72252 C59WMP 118724020 IC50 = 330.1 nM T72252 C7ZJL3 118724021 IC50 = 198.3 nM T72252 CG47EC 118724022 IC50 = 111.9 nM T72252 CJ6M2B 118724023 IC50 = 109 nM T72252 CNPQ61 118724024 IC50 = 72.5 nM T72252 CAWQ46 118724025 IC50 = 63.7 nM T72252 CM51UC 118724026 IC50 = 86.9 nM T72252 CO3J7G 118724027 IC50 = 78.4 nM T72252 CJ4F9Q 118724028 IC50 = 59.7 nM T72252 CN8A0V 118724029 IC50 = 158.2 nM T72252 C8TAO7 118724030 IC50 = 72.7 nM T72252 CP2QC1 118724031 IC50 = 166.3 nM T72252 CN5WS2 118724032 IC50 = 97.9 nM T72252 CXN5D4 118724033 IC50 = 74.9 nM T72252 CXZ70W 118724034 IC50 = 100.9 nM T72252 CQ68TB 118724035 IC50 = 18080 nM T72252 CJC7S1 118724036 IC50 = 56.7 nM T72252 CMN80F 118724037 IC50 = 115.1 nM T72252 CBNT42 118724038 IC50 = 115 nM T72252 C5S2MJ 118724039 IC50 = 296.7 nM T72252 CEB4O2 118724040 IC50 = 185.1 nM T72252 C9QKI3 127020966 IC50 > 100000 nM T72252 CWM2E8 133081971 IC50 > 9999 nM T72252 CLDI36 137225012 IC50 > 200000 nM T72252 C17RCJ 137225013 IC50 > 200000 nM T72252 C4H1LQ 137225014 IC50 > 200000 nM T72252 C0J4OC 137225015 IC50 > 200000 nM T72252 CW41CO 137225056 IC50 > 200000 nM T72252 C7D4QS 137225083 IC50 > 200000 nM T72252 C7UFH6 137225092 IC50 > 200000 nM T72252 CU42CE 155567829 IC50 > 100000 nM T72252 D0L9AX 644345 IC50 = 59.1 nM T72252 D0N5MU 4117381 Ki = 3000 nM T72252 D0Q9XX 515950 Ki = 290 nM T72252 D0V6DX 10640 IC50 = 386 nM T72252 D0Y5IQ 44255320 IC50 = 5000 nM T40098 C5O9HZ 18960776 IC50 = 600 nM T40098 CQ18BI 56643478 IC50 > 30000 nM T40098 C7N1QX 56658802 IC50 = 25000 nM T40098 C20AZO 56658809 IC50 = 2900 nM T40098 CT7CQ2 56658922 IC50 = 7000 nM T40098 CDCU98 56658927 IC50 = 7400 nM T40098 CT05HU 56658938 IC50 = 1900 nM T40098 CB7T3O 56662138 IC50 = 3900 nM T40098 CA2J4M 56665726 IC50 = 810 nM T40098 C8JQW7 56665736 IC50 = 1000 nM T40098 CIM4P9 56665873 IC50 = 1400 nM T40098 CPXA70 56668892 IC50 = 1800 nM T40098 C6WEH2 56669055 IC50 = 7600 nM T40098 CQD5C8 56669167 IC50 = 1900 nM T40098 CTSQ34 56669318 IC50 = 4400 nM T40098 CD06RX 56672370 IC50 = 1300 nM T40098 CT63HW 56672642 IC50 = 3600 nM T40098 CCRS13 56672791 IC50 = 300 nM T40098 CMF08O 56672796 IC50 = 2600 nM T40098 CNH9V6 56675904 IC50 = 2300 nM T40098 C03UBX 56676113 IC50 = 1900 nM T40098 C0V2RQ 56676125 IC50 = 1000 nM T40098 C8HG7I 56676130 IC50 = 3900 nM T40098 CH8M0Y 56679074 IC50 = 1100 nM T40098 C8J7BN 56679210 IC50 = 1400 nM T40098 CTVO23 56679447 IC50 = 900 nM T40098 CB4KV6 56682374 IC50 = 4100 nM T40098 CO08CN 56682503 IC50 = 5000 nM T40098 C6HGP3 56682632 IC50 = 3900 nM T40098 C0ICP9 56682640 IC50 = 6900 nM T40098 CIK8W1 56682645 IC50 = 5600 nM T40098 C02ISO 71583406 IC50 = 2800 nM T40098 CBI6Z7 71583526 IC50 = 600 nM T40098 CE1RQ2 71817009 IC50 > 50000 nM T40098 CPW95C 71817013 IC50 > 50000 nM T40098 C0CLR8 71817014 IC50 > 50000 nM T40098 CO27TU 71817052 IC50 > 50000 nM T40098 CDF47R 71817054 IC50 > 50000 nM T40098 C4VJU6 71817055 IC50 > 50000 nM T40098 C95KPI 71817090 IC50 > 50000 nM T40098 C1UK4V 71817091 IC50 > 50000 nM T40098 CZ83QK 145960490 IC50 > 50000 nM T40098 C2J9YV 154727580 IC50 = 128000 nM T40098 CDV4Z6 155515709 IC50 = 766000 nM T31479 D0K8KX 5280343 IC50 = 2000 nM T31479 D00XQO 6437368 IC50 = 3900 nM T31479 CK7IR6 155815 IC50 = 228 nM T31479 CBNC27 9801919 IC50 = 3 nM T31479 CU79BR 9801920 IC50 = 390 nM T31479 CFB7V6 9802744 IC50 = 5 nM T31479 C1BS0W 9803388 IC50 = 364 nM T31479 CO3M2Q 9803692 IC50 = 3 nM T31479 CWS9O0 9846179 IC50 = 1090 nM T31479 CZSL21 9847448 IC50 = 6 nM T31479 CA6W3U 9863966 IC50 = 761 nM T31479 C23IEK 9866653 IC50 = 800 nM T31479 C3QI5S 9867345 IC50 = 84 nM T31479 C2S6FM 9869328 IC50 = 130 nM T31479 C3LMS6 9869329 IC50 = 17 nM T31479 C78TJF 9886168 IC50 = 5 nM T31479 C20UBZ 9888132 IC50 = 1200 nM T31479 CZ4UP6 9911907 IC50 = 3 nM T31479 C9BW4J 9955004 IC50 = 570 nM T31479 CFE12L 9958280 IC50 > 1600 nM T31479 C7W6GZ 10016808 IC50 = 6200 nM T31479 CE3H0R 10187432 IC50 > 1600 nM T31479 CB53QZ 10223158 IC50 > 1600 nM T31479 C12IMN 10389981 IC50 = 1.3 nM T31479 CX8QO3 10403265 IC50 = 9500 nM T31479 C50IKB 10406575 IC50 = 3 nM T31479 CFZ59K 10435114 IC50 = 10000 nM T31479 CZ89RL 10509638 IC50 = 90000000 nM T31479 CD7V9Z 10524659 IC50 = 51 nM T31479 C2EKY3 10528351 IC50 = 62 nM T31479 CF73HI 10528864 IC50 = 35 nM T31479 C27VMJ 10530468 IC50 = 55000 nM T31479 C1ZIT8 10546433 IC50 = 62 nM T31479 C91AKI 10549423 IC50 = 51 nM T31479 CKS7W5 10550293 IC50 = 36 nM T31479 CXWN27 10551187 IC50 = 14 nM T31479 CEB1F4 10558196 IC50 = 9000000 nM T31479 CU1O7K 10574655 IC50 = 7.3 nM T31479 CRX18G 10576315 IC50 = 240 nM T31479 CIAX35 10596664 IC50 = 49 nM T31479 CQM42R 10597121 IC50 = 23 nM T31479 C1TP0V 10597576 IC50 > 50000 nM T31479 C3ZK9R 10598416 IC50 = 120 nM T31479 CPK1L8 10599954 IC50 = 13 nM T31479 CP3EQ6 10601203 IC50 = 6600 nM T31479 CAP0M4 10620165 IC50 = 11 nM T31479 C3PLX0 10620311 IC50 = 780 nM T31479 C0IZ5H 10624196 IC50 = 4.2 nM T31479 CD1P2G 10624896 IC50 = 83 nM T31479 CMX52V 10625527 IC50 = 280 nM T31479 CR5Q8G 10642134 IC50 = 14 nM T31479 C3G7JS 10643736 IC50 = 29 nM T31479 C69WSI 10643875 IC50 = 21 nM T31479 CEX2O5 10645128 IC50 = 1100 nM T31479 CLD27J 10647376 IC50 = 26 nM T31479 C79XPV 10648564 IC50 = 80 nM T31479 C6PWL8 10666992 IC50 = 19 nM T31479 C8HYP0 10669802 IC50 = 38 nM T31479 CL6PS3 10671490 IC50 = 1.4 nM T31479 C2SVD1 10672182 IC50 = 16 nM T31479 C2WAN3 10672505 IC50 = 140 nM T31479 CJ4XR6 10694211 IC50 = 5 nM T31479 C6S8OH 10723410 IC50 > 100000000 nM T31479 CGLW34 10742448 IC50 = 13 nM T31479 C32NEP 10761796 IC50 = 10 nM T31479 CZ8E1T 10767354 IC50 = 46 nM T31479 C6N1GO 10784865 IC50 > 100000 nM T31479 CEO1Y4 10784983 IC50 > 100000 nM T31479 CC91UG 10786795 IC50 > 50000 nM T31479 CJ0L7E 10786797 IC50 = 80 nM T31479 CI52FX 10811610 IC50 = 43 nM T31479 CTD1F8 10813678 IC50 = 1400 nM T31479 CS60RI 10813679 IC50 = 23 nM T31479 CP8B4O 10815184 IC50 = 100 nM T31479 CO57ZR 10835629 IC50 = 19000 nM T31479 C9O7KE 10842569 IC50 > 100000000 nM T31479 CW0F3K 10843834 IC50 = 11000000 nM T31479 CHG89F 10865991 IC50 = 135000000 nM T31479 C56AIM 11610604 IC50 = 2000 nM T31479 CW65ZB 11726406 IC50 = 13 nM T31479 CKM92O 11795292 IC50 = 15 nM T31479 CP5I4L 11795826 IC50 = 30 nM T31479 C0KBW4 12114490 IC50 = 4400 nM T31479 CE02QD 15250860 IC50 = 13800 nM T31479 C8T0ER 16135012 IC50 = 18000000 nM T31479 CS59WD 16138504 IC50 = 55000000 nM T31479 CPS02Y 16143405 IC50 = 6500000 nM T31479 CW09CU 16144090 IC50 > 100000000 nM T31479 CS8LO6 16144962 IC50 > 100000000 nM T31479 CE89KY 16157140 IC50 = 6600000 nM T31479 CG1Y0D 20592756 IC50 = 200 nM T31479 CK5G0Z 20592757 IC50 = 3400 nM T31479 C4F7TS 20644949 IC50 > 1600 nM T31479 C2KVQ7 21585456 IC50 = 21500 nM T31479 C05YWA 21774719 IC50 = 3700 nM T31479 CR9T8M 24950865 IC50 = 1300 nM T31479 CW14ZE 24950866 IC50 > 1600 nM T31479 CJD2K3 24950867 IC50 = 1400 nM T31479 CLTX47 24951184 IC50 = 810 nM T31479 C7HON4 24951342 IC50 > 1600 nM T31479 CE1W6P 44343949 IC50 = 5300 nM T31479 CHD2O0 44343951 IC50 = 31000 nM T31479 C76ALP 44346729 IC50 > 50000 nM T31479 C9G7TK 44346748 IC50 > 50000 nM T31479 C53ZRT 44346872 IC50 = 15000000 nM T31479 CNC97E 44346890 IC50 = 12000000 nM T31479 CJVF24 44346894 IC50 = 170000 nM T31479 C0UQJ9 44346921 IC50 = 200000 nM T31479 CDL62X 44346946 IC50 = 25000 nM T31479 CO76RA 44346948 IC50 = 67000 nM T31479 CF4WT5 44346961 IC50 = 17 nM T31479 CMV46D 44346973 IC50 = 400000 nM T31479 CM57HR 44346974 IC50 = 100000 nM T31479 CFTP94 44347129 IC50 = 1300 nM T31479 C84VUD 44347150 IC50 = 7000 nM T31479 CI63SR 44347181 IC50 = 240000 nM T31479 CF97EX 44347250 IC50 = 910000 nM T31479 CBJR09 44347264 IC50 = 160000 nM T31479 CF78XL 44347265 IC50 = 420000 nM T31479 CNBD26 44347266 IC50 = 45000 nM T31479 CZF0U8 44347291 IC50 = 30 nM T31479 CJH4G6 44347353 IC50 = 20 nM T31479 C5V7RS 44347355 IC50 = 11 nM T31479 CS6CM0 44347418 IC50 = 22000 nM T31479 CEH6I0 44347419 IC50 = 80 nM T31479 CWA42C 44365795 IC50 > 100000000 nM T31479 CLBM81 44365796 IC50 = 100000000 nM T31479 C0PBQ3 44365926 IC50 > 100000000 nM T31479 CFRO56 44365927 IC50 = 60000000 nM T31479 C7R5LV 44365928 IC50 = 100000000 nM T31479 CY79AC 44365929 IC50 > 100000000 nM T31479 C81GRO 44568005 IC50 = 36000 nM T31479 CLD4I9 44578597 IC50 > 1600 nM T31479 C9CY8T 44583739 IC50 = 3800 nM T31479 C2EGY0 76331562 IC50 = 98000000 nM T31479 CF32QE 122197354 IC50 = 10000000 nM T31479 C1VB6C 122197355 IC50 = 60000000 nM T31479 C2PU7S 122197356 IC50 > 100000000 nM T31479 C6C2FI 135540837 IC50 > 100000 nM T31479 C5FZ1G 135540866 IC50 = 10000 nM T31479 CHZP29 135540867 IC50 = 15000 nM T31479 CUL9R8 135540870 IC50 = 18000 nM T31479 CABE48 135589918 IC50 = 5750 nM T31479 CQO58C 135993329 IC50 = 7600 nM T31479 C9LI3K 135993330 IC50 = 8700 nM T31479 D05DUX 17748437 IC50 = 1600 nM T31479 D0H1JX 10362969 IC50 = 3000 nM T31479 D0L3IQ 442153 IC50 = 6000 nM T31479 D0SJ2Q 10494 IC50 = 3000 nM T86552 C0C7MF 641818 IC50 = 14000 nM T86552 C04TZH 917172 IC50 = 3400 nM T86552 C5HW9C 3631514 IC50 = 130 nM T86552 C9ALF1 3641989 IC50 = 4500 nM T86552 CU20KN 4449347 IC50 = 14100 nM T86552 CM85RB 5286094 IC50 = 25000 nM T86552 CE80AQ 5327044 IC50 = 22000 nM T86552 CY5A9Z 5350510 IC50 = 29000 nM T86552 C3SVB9 5712095 IC50 = 15000 nM T86552 CCAT78 5723044 IC50 = 6000 nM T86552 CY04US 5850698 IC50 = 47000 nM T86552 C5PS1Z 5998054 IC50 = 1000 nM T86552 CW16CY 6017999 IC50 = 6000 nM T86552 CFO1R0 6063342 IC50 = 7000 nM T86552 C0WT5I 6065576 IC50 = 8000 nM T86552 C32KUP 6091793 IC50 > 50000 nM T86552 CX7LK3 9891755 IC50 = 5000 nM T86552 CFO76R 10413405 IC50 = 1000 nM T86552 CE9Z6D 18171887 IC50 = 8000 nM T86552 C0VIM7 18171890 IC50 = 3000 nM T86552 CN13PF 18171892 IC50 = 3000 nM T86552 C52UYZ 21041603 IC50 = 1000 nM T86552 CJ0AH9 21041609 IC50 = 17000 nM T86552 CWD08Q 22025531 IC50 = 1000 nM T86552 CO25NE 22025534 IC50 = 5000 nM T86552 CX09FH 22025535 IC50 = 3000 nM T86552 CWE71Q 22025537 IC50 = 3000 nM T86552 C6DJP4 22025539 IC50 = 7000 nM T86552 C7IFR3 22025540 IC50 = 3000 nM T86552 CI76OG 22025542 IC50 = 2000 nM T86552 CXO3G1 22025544 IC50 = 11000 nM T86552 CVM98W 22025545 IC50 = 2000 nM T86552 C5U2ST 22025548 IC50 = 6000 nM T86552 CF7NO6 22025549 IC50 = 2000 nM T86552 C8R4HX 22025550 IC50 = 2000 nM T86552 C5GMD4 22025552 IC50 = 12000 nM T86552 CJHP63 22025555 IC50 = 2000 nM T86552 CH17PY 22025558 IC50 = 3000 nM T86552 CHJ3E2 22025560 IC50 = 2000 nM T86552 C5R4QB 22025562 IC50 = 2000 nM T86552 CYSX31 22025563 IC50 = 4000 nM T86552 CJ5R7P 22025564 IC50 = 4000 nM T86552 CQ34JS 22025565 IC50 = 3000 nM T86552 CO9I2H 22025566 IC50 = 7000 nM T86552 C7K6MB 22025568 IC50 = 4000 nM T86552 COPV18 22025571 IC50 = 2000 nM T86552 C0UF5S 22025572 IC50 = 4000 nM T86552 CB5KY9 22025573 IC50 = 2000 nM T86552 C9U8KM 22025576 IC50 = 2000 nM T86552 CN1M9U 22025578 IC50 = 4000 nM T86552 C2AUJ3 22025583 IC50 = 3000 nM T86552 C0J9YM 22025587 IC50 = 3000 nM T86552 CIR46G 22025589 IC50 = 3000 nM T86552 CU9WV7 44284440 IC50 = 4000 nM T86552 CN3XF6 44284588 IC50 = 5000 nM T86552 C2DT0H 44284622 IC50 > 50000 nM T86552 CM0V8K 44284625 IC50 = 15000 nM T86552 CF6H4R 44284630 IC50 = 2000 nM T86552 CU6F5N 44284664 IC50 = 2000 nM T86552 COM5R1 44284668 IC50 > 50000 nM T86552 C1IT9N 44284712 IC50 = 17000 nM T86552 C4EIA5 44284714 IC50 = 9000 nM T86552 C8PHW9 44284788 IC50 = 4000 nM T86552 CI8K9R 44284791 IC50 = 3000 nM T86552 CON5Y6 44284792 IC50 = 5000 nM T86552 C9MN2O 44284793 IC50 = 3000 nM T86552 CFE7J8 44284819 IC50 = 4000 nM T86552 CBW7C4 44284834 IC50 = 2000 nM T86552 C6QH3N 44284836 IC50 = 3000 nM T86552 C5FNC9 44284843 IC50 = 3000 nM T86552 CZKF34 44284899 IC50 = 2000 nM T86552 CA1FL3 44284901 IC50 = 3000 nM T86552 CGV0U1 44284902 IC50 > 50000 nM T86552 CQ4X2D 44284903 IC50 > 50000 nM T86552 C4E6ST 44284904 IC50 = 2000 nM T86552 CX48LT 44284923 IC50 = 4000 nM T86552 CMEQ96 44284944 IC50 = 1000 nM T86552 CX0K1Z 44284964 IC50 = 4000 nM T86552 C7ZT3E 44285090 IC50 = 6000 nM T86552 CV3UC2 44285094 IC50 > 50000 nM T86552 CM4AE5 44285106 IC50 = 1000 nM T86552 C46HCU 44285107 IC50 = 1000 nM T86552 C0LIY6 44285165 IC50 = 1000 nM T86552 C86GHF 44366282 IC50 = 780 nM T86552 C1N8KY 44366424 IC50 = 390 nM T86552 C12EBC 44366437 IC50 = 670 nM T86552 C3R4JO 44366441 IC50 = 280 nM T86552 CN96WU 44366472 IC50 = 310 nM T86552 CF39TX 44366481 IC50 = 1900 nM T86552 C75QDR 44366482 IC50 = 1000 nM T86552 C4G7ZA 44366518 IC50 = 320 nM T86552 CN90PO 44366776 IC50 = 610 nM T86552 CDA2V8 44366837 IC50 = 2800 nM T86552 CC3JQ2 44366838 IC50 = 300 nM T86552 CG2D0J 44366849 IC50 = 11000 nM T86552 CO90MY 44366867 IC50 = 2000 nM T86552 CXQ2K9 44367057 IC50 = 280 nM T86552 CGP1T4 44367072 IC50 = 140 nM T86552 CHW3A0 44367073 IC50 = 40000 nM T86552 C1ULK2 44367098 IC50 = 1700 nM T86552 CD1TA0 44367101 IC50 = 2100 nM T86552 C3HW7L 44570553 IC50 = 2000 nM T86552 C17PVE 44570554 IC50 = 13000 nM T86552 CLOY92 44570599 IC50 = 20000 nM T86552 CK06LT 44570600 IC50 = 5000 nM T86552 C7LER5 73669500 IC50 > 31000 nM T86552 CJKB83 73670174 IC50 > 31000 nM T86552 CS72RV 117885758 IC50 > 31000 nM T86552 C6Z3NJ 117885766 IC50 > 31000 nM T86552 CKU6S4 117885912 IC50 > 31000 nM T86552 CR7DJ0 118453722 IC50 > 31000 nM T86552 CK1Z7I 118462026 IC50 > 31000 nM T86552 CC53OH 135403101 IC50 = 1800 nM T86552 CAT93B 135421580 IC50 = 790 nM T86552 C2CQB3 135457340 IC50 = 1000 nM T86552 CZHL28 135478288 IC50 = 13000 nM T86552 CI14OR 135921196 IC50 = 400 nM T86552 C25SZC 135921197 IC50 = 600 nM T86552 C7MKR6 135921198 IC50 = 5500 nM T86552 CPW15D 136094894 IC50 = 10200 nM T86552 CGK05C 145965353 IC50 = 770 nM T86552 D06ERH 637760 IC50 = 23000 nM T97589 D02UFQ 11620908 IC50 > 10000 nM T97589 D0E3TC 44259 IC50 = 19.9 nM T97589 D0RN3S 71245288 IC50 = 6 nM T97589 D03BNU 59604787 IC50 > 10000 nM T97589 D0T3ME 156422 IC50 > 30000 nM T97589 C7VH4Q 70976 IC50 = 13300 nM T97589 C39NYX 71029 IC50 > 10000 nM T97589 CCS9M8 650462 IC50 = 25000 nM T97589 CJWL84 712714 IC50 = 10000 nM T97589 CF1I8A 756688 IC50 = 25800 nM T97589 CRG4L5 793884 IC50 = 4700 nM T97589 CCB42L 836391 IC50 = 260 nM T97589 CWNF57 1201118 IC50 > 33000 nM T97589 CRVD70 1201167 IC50 > 33000 nM T97589 C8MXI1 1205453 IC50 = 1250 nM T97589 CI2C6M 1205717 IC50 = 750 nM T97589 CL2H9X 1207357 IC50 > 33000 nM T97589 C80SLR 1351628 IC50 = 200 nM T97589 C5FN9Z 1351934 IC50 = 350 nM T97589 CD8F2Z 1368457 IC50 = 1000 nM T97589 CF1A5C 1377508 IC50 > 33000 nM T97589 C7X6NE 1420181 IC50 > 33000 nM T97589 CZCR37 1544033 IC50 = 300 nM T97589 C5RS0G 1549274 IC50 > 10000 nM T97589 CNB34V 1587088 IC50 = 2000 nM T97589 C9RW2G 1589300 IC50 = 500 nM T97589 CB30VG 1589310 IC50 = 200 nM T97589 CSHB27 1589389 IC50 = 350 nM T97589 CJQ25S 1591868 IC50 > 33000 nM T97589 CE6DC8 1594457 IC50 > 33000 nM T97589 CKY7T2 1602082 IC50 = 35000 nM T97589 CW6P1V 1636949 IC50 > 33000 nM T97589 CZ3TU2 1641056 IC50 = 650 nM T97589 CENS71 2261810 IC50 > 33000 nM T97589 CCUF19 2942922 IC50 = 42600 nM T97589 CABJ52 3129049 IC50 = 17000 nM T97589 CW02ZH 3384409 IC50 = 35500 nM T97589 C4VFQ8 3408837 IC50 = 4500 nM T97589 CF37SN 3466082 IC50 = 38000 nM T97589 CA05SH 3510382 IC50 = 28200 nM T97589 CBC19W 3530671 IC50 = 1550 nM T97589 C0V8RG 3605180 IC50 = 2000 nM T97589 CZ86DH 3619463 IC50 = 4400 nM T97589 CIJ48H 3777223 IC50 = 31000 nM T97589 CZ5BL1 3793962 IC50 = 29500 nM T97589 CWS43T 3811046 IC50 = 63000 nM T97589 CH63SV 3811406 IC50 = 30200 nM T97589 C8AM4K 3839807 IC50 = 4200 nM T97589 CQH47Z 3845066 IC50 = 28200 nM T97589 CL9NE8 3953315 IC50 = 28200 nM T97589 C85ANT 4271048 IC50 = 9100 nM T97589 CESD45 5522952 Ki = 500 nM T97589 C7NSH6 5827971 IC50 = 500 nM T97589 C9V5GK 5828227 IC50 = 500 nM T97589 C24XJT 5828229 IC50 = 1000 nM T97589 CV7S6O 5941094 IC50 = 2800 nM T97589 CUH30G 6064827 IC50 = 300 nM T97589 CVZG21 6157349 IC50 = 2000 nM T97589 CRS19W 6197516 IC50 = 3600 nM T97589 CX7PY1 6206672 IC50 > 33000 nM T97589 CH4W8C 6275433 IC50 = 2500 nM T97589 C8OV5P 6275436 IC50 = 5000 nM T97589 CI0N6L 6275437 IC50 = 5200 nM T97589 C5ZCG8 6275597 IC50 = 4600 nM T97589 C6FJ5R 6275602 IC50 = 5200 nM T97589 CI6LK1 6509437 IC50 = 1800 nM T97589 C4KIM7 6509439 Ki = 340 nM T97589 CH1ZN6 6516664 IC50 = 500 nM T97589 CR5YT8 7454869 IC50 = 3000 nM T97589 CAC5D7 7454873 IC50 = 3000 nM T97589 CPE97D 9878655 IC50 = 82700 nM T97589 CN3HY4 12413939 IC50 > 10000 nM T97589 CPGW52 16086083 IC50 > 10000 nM T97589 CL16IH 16271725 IC50 = 1800 nM T97589 CFZ2S4 16422835 IC50 = 18900 nM T97589 CGL54Y 16446616 IC50 = 750 nM T97589 C4TKL8 16446617 IC50 = 520 nM T97589 CA9M7G 17881853 IC50 > 10000 nM T97589 CRX6H4 23474918 IC50 = 750 nM T97589 CY8L7E 24896769 IC50 > 10000 nM T97589 CQ5V7O 24944928 IC50 = 32 nM T97589 CLG1H8 24945008 IC50 = 6.3 nM T97589 CJA06T 25118862 IC50 = 251 nM T97589 C02OPU 39354723 IC50 > 10000 nM T97589 CF6S3O 43861157 IC50 > 33000 nM T97589 CEL61X 44229839 IC50 > 10000 nM T97589 C3VRO9 44557921 IC50 > 10000 nM T97589 C4SE6K 44786797 IC50 = 3900 nM T97589 C2MI6X 44786879 IC50 = 750 nM T97589 C5C3YT 44786880 IC50 = 500 nM T97589 CU21XL 44786881 IC50 = 500 nM T97589 CZ58FY 46215814 IC50 = 5690 nM T97589 CAL7Y8 53319927 IC50 = 15 nM T97589 C0GB8U 53321232 IC50 = 19 nM T97589 C8NA4L 53384644 IC50 > 30000 nM T97589 CN9QD7 56643097 IC50 > 10000 nM T97589 C8BO7K 56644085 IC50 = 18 nM T97589 C62DCN 56644086 IC50 = 9 nM T97589 CCBQ25 59175229 IC50 = 22 nM T97589 CR0J1M 59175292 IC50 = 21 nM T97589 CDG1W3 59175319 IC50 = 82 nM T97589 C8I6KT 59175417 IC50 = 21 nM T97589 CSO56Y 59175418 IC50 = 870 nM T97589 CE8WC4 59175460 IC50 = 129 nM T97589 C5Y0KL 59175469 IC50 = 70 nM T97589 CZ6NB4 59175598 IC50 = 30 nM T97589 CBH5K0 59175648 IC50 = 34 nM T97589 CT2N8Z 59175651 IC50 = 16 nM T97589 CV63UL 67240318 IC50 > 10000 nM T97589 CB7QV0 68603188 IC50 > 10000 nM T97589 CEBO91 71452977 IC50 > 10000 nM T97589 C2JZV1 71578449 IC50 > 33000 nM T97589 C7OKB8 71578450 IC50 > 33000 nM T97589 C36BJZ 71581421 IC50 = 251 nM T97589 CD15HJ 71581422 IC50 = 50 nM T97589 CB1GH4 71581423 IC50 = 7.9 nM T97589 CZ31PU 71583657 IC50 > 10000 nM T97589 CSNR61 71716557 IC50 = 2500 nM T97589 C4WIL9 71718392 IC50 = 800 nM T97589 C9XK6B 89070277 IC50 > 10000 nM T97589 C5CPX7 89070280 IC50 > 10000 nM T97589 C1ZFC6 90231952 IC50 = 0.7 nM T97589 C0Y8ZK 91933875 IC50 > 1000 nM T97589 C19INJ 117091972 IC50 = 2000 nM T97589 CT56BP 118729143 IC50 = 4200 nM T97589 CN0UF9 118729144 IC50 = 5000 nM T97589 CMB52T 118729145 IC50 = 2000 nM T97589 CY23GB 118729146 IC50 = 4400 nM T97589 CUX8G2 118729147 IC50 = 7600 nM T97589 CG4TA8 118729148 IC50 = 2900 nM T97589 C6KR4J 118729149 IC50 = 5500 nM T97589 CRLH90 118729150 IC50 = 6300 nM T97589 CFM57X 118729151 IC50 = 17000 nM T97589 C29KJL 124222752 IC50 = 400 nM T97589 CDQU61 127053598 EC50 = 6.31 nM T97589 CY2A0O 127053601 IC50 = 5.012 nM T97589 CL6UK9 127053602 IC50 = 12.59 nM T97589 CN08AJ 131955124 IC50 = 1.5 nM T97589 CWNA90 131955125 IC50 = 2.4 nM T97589 CMUY57 134136917 IC50 = 50.12 nM T97589 C4M8IZ 134137100 IC50 = 50.12 nM T97589 CVY03I 134137951 IC50 = 31.62 nM T97589 C3QOF5 134140640 IC50 = 19.95 nM T97589 C80FHO 134141475 IC50 = 12.59 nM T97589 CFN83Y 134144068 IC50 = 794.33 nM T97589 C6OM5U 134145185 IC50 = 39.81 nM T97589 CV7SN1 134145495 IC50 = 19.95 nM T97589 CS1H6B 134149289 IC50 = 15.85 nM T97589 C1XT4K 134150112 EC50 = 15.85 nM T97589 C7NI5Z 134152962 EC50 = 12.59 nM T97589 C8P6RH 134154870 IC50 = 398.11 nM T97589 CG0OP9 134155797 IC50 = 10 nM T97589 CL7F8K 134157323 IC50 = 6000 nM T97589 C54FXD 134957362 IC50 > 10000 nM T97589 C80QXW 135423664 IC50 = 15000 nM T97589 CF15TS 135477211 IC50 = 35000 nM T97589 CK58TZ 137635507 IC50 = 100000 nM T97589 CVEK25 137636074 EC50 = 140 nM T97589 C7TG3J 137641313 EC50 = 60 nM T97589 CPL9Q1 137644068 EC50 = 99 nM T97589 CQ7Y2I 137646649 EC50 = 130 nM T97589 CFE92C 137647290 EC50 = 600 nM T97589 CL0H5M 137648830 IC50 = 500000 nM T97589 CQ3M7P 137655650 EC50 = 65 nM T97589 C3HT7D 138458386 IC50 = 4 nM T97589 C2ZQ0L 138458432 IC50 <= 100 nM T97589 CJ16FS 138458448 IC50 = 25 nM T97589 C9P5LC 138458561 IC50 = 31 nM T97589 C7I4YZ 138458674 IC50 = 658 nM T97589 C2OCB0 139589936 IC50 > 50000 nM T97589 C2W4NJ 139589937 IC50 = 740 nM T97589 CK90DE 139589938 IC50 > 50000 nM T97589 C1OXF6 139589939 IC50 = 3000 nM T97589 C0NCJ7 139589940 IC50 > 50000 nM T97589 CNW73T 139589941 IC50 = 6400 nM T97589 C1PVA9 139589942 IC50 = 1100 nM T97589 CO73YE 139589944 IC50 = 4100 nM T97589 CAKT08 140430627 IC50 = 4 nM T97589 C1VUO5 142411816 IC50 = 165 nM T97589 CP73TY 142411827 IC50 = 6 nM T97589 C08WOT 142411831 IC50 <= 100 nM T97589 CZI8D0 142411860 IC50 <= 100 nM T97589 CG1KI6 142411901 IC50 <= 100 nM T97589 C06TLE 142411916 IC50 = 1437 nM T97589 CO7R5P 142411943 IC50 = 100 nM T97589 CQX6Y2 142411956 IC50 = 43 nM T97589 CZ0L5V 142411973 IC50 = 8 nM T97589 C5X7ZV 142411981 IC50 = 28 nM T97589 CH3P7D 142411991 IC50 = 350 nM T97589 C4PYK9 142412044 IC50 = 11 nM T97589 CN34ST 142412072 IC50 <= 100 nM T97589 C6VB3O 145925651 IC50 >= 5000 nM T97589 CWLQ39 145963899 IC50 = 900 nM T97589 CB4V8Y 145964189 IC50 > 10000 nM T97589 C0GI2D 145964450 IC50 > 10000 nM T97589 C50CYG 145967046 IC50 > 10000 nM T97589 C16QTH 145967480 IC50 > 10000 nM T97589 CH34CK 145971544 IC50 > 10000 nM T97589 C1PIV2 145971548 IC50 > 10000 nM T97589 CYDI91 145972315 IC50 > 10000 nM T97589 CQ3VL2 145973695 IC50 = 200 nM T97589 CP2N4K 145974025 IC50 = 600 nM T97589 CXZ08M 145974364 IC50 > 10000 nM T97589 CMF07J 145975267 IC50 > 10000 nM T97589 C5FQU2 145975617 IC50 > 10000 nM T97589 CU7I9D 145977879 IC50 > 10000 nM T97589 CE5ZW0 145978186 IC50 > 10000 nM T97589 C0O4NB 145978703 IC50 > 10000 nM T97589 C89TSV 145981571 IC50 = 1 nM T97589 CP97BA 145982455 IC50 = 770 nM T97589 C6UW9H 145986328 IC50 = 4 nM T97589 C1BW6I 145989111 IC50 = 0.32 nM T97589 C1BC3Q 145990004 IC50 = 170 nM T97589 CKO81L 145990765 IC50 = 0.1 nM T97589 C1RLD9 145990863 IC50 = 73 nM T97589 CIU0W6 145991814 IC50 = 140 nM T97589 CSD6W8 145993521 IC50 = 580 nM T97589 C7FD2A 145994100 IC50 = 0.42 nM T97589 C2MD1Q 155513187 IC50 > 10000 nM T97589 CXIK13 155521986 IC50 = 76 nM T97589 CN17LD 155529041 IC50 = 14 nM T97589 CLK08R 155534100 IC50 = 161 nM T97589 C2CG1A 155537016 IC50 > 10000 nM T97589 C4G2FA 155542760 IC50 = 92 nM T97589 C7LXR5 155551184 IC50 = 8 nM T97589 C23AUN 155555164 IC50 = 299 nM T97589 CL7Q4P 155568326 IC50 = 8 nM T97589 D01WIH 51998 IC50 > 10000 nM T97589 D0EU1R 46215815 IC50 > 27542 nM T97589 D0F0AX 135413546 IC50 = 7000 nM T97589 D0F0XZ 25214468 IC50 = 13 nM T97589 D0Q0YV 24944925 IC50 = 14 nM T97589 D0R1FT 4564 IC50 = 25100 nM T64725 D0S0RS 24988881 IC50 > 100000000 nM T64725 C2GVL4 15980639 IC50 > 100000000 nM T64725 C1VQZ8 15980754 IC50 > 2000 nM T64725 C13RAO 16042458 IC50 > 100000000 nM T64725 CX28KD 24988880 IC50 > 100000000 nM T64725 CV6UH1 25167051 IC50 > 20000 nM T64725 CP6K5Q 46916548 IC50 > 80000 nM T64725 C9S6NM 53388366 IC50 > 100000000 nM T64725 D0O3TT 11973722 IC50 > 10000 nM T99799 D04AIT 5280445 Ki = 166100 nM T99799 D06OMW 3052776 IC50 = 4760 nM T99799 D06XWB 854026 IC50 > 100000 nM T99799 D07XYV 54766 IC50 = 3 nM T99799 D08USJ 4456 IC50 = 16300 nM T99799 D09QDP 4380 IC50 > 500000 nM T99799 D09QEI 4740 IC50 > 50000 nM T99799 D0B3HD 2519 IC50 > 50000 nM T99799 D0E6YQ 1935 IC50 = 0.9 nM T99799 D0K8KX 5280343 Ki = 68000 nM T99799 D0L4JT 5333 IC50 = 138790 nM T99799 D0NS6H 3152 IC50 = 14 nM T99799 D0O2WB 4991 IC50 = 900 nM T99799 D0Q0RC 3290 Ki = 20 nM T99799 D0R1QE 3672 IC50 < 600000 nM T99799 D0R9VR 9651 IC50 = 0.38 ug.mL-1 T99799 D0S2UG 26757 IC50 > 500000 nM T99799 D0UU9Y 4938 IC50 > 50000 nM T99799 D0W8WB 2353 IC50 = 1090 nM T99799 D0WY5Q 77991 IC50 = 30 nM T99799 D01LYX 65872 IC50 = 0.69 nM T99799 D02EVF 6112 IC50 > 1000000 nM T99799 D07CIN 192706 IC50 = 1560 nM T99799 D07SDQ 969516 IC50 > 5000 nM T99799 D0B1FE 3194 IC50 = 4600 nM T99799 D0B6IZ 137905 Ki > 100000 nM T99799 D0M3IN 1188 IC50 > 50000 nM T99799 D0U3EP 445154 IC50 > 5000 nM T99799 D09JVV 5983 IC50 = 15 nM T99799 D0B2BQ 135462830 IC50 = 7200 nM T99799 D0S1VV 119053 IC50 = 21000 nM T99799 CXU4W0 650 Ki > 100000 nM T99799 CT6RA0 2317 IC50 = 6165.95 nM T99799 C0RFA2 3102 Ki > 100000 nM T99799 C8F5QC 5077 IC50 = 11000 nM T99799 C8GZO5 5741 IC50 = 7273 nM T99799 CKB56J 5824 IC50 = 60 nM T99799 CX82HQ 6070 IC50 = 19460 nM T99799 C4IU5T 6889 Ki > 100000 nM T99799 C5NIV3 7088 IC50 = 19200 nM T99799 C5EUF4 7108 IC50 = 5800 nM T99799 C6NQ4X 8246 IC50 = 800 nM T99799 CJL02I 8307 IC50 = 1370000 nM T99799 CTY1W5 9820 Ki = 50 nM T99799 C25CYL 10434 Ki > 100000 nM T99799 C47FYB 10662 Ki > 100000 nM T99799 C2G5AW 11066 IC50 = 68000 nM T99799 COGY52 11321 Ki > 100000 nM T99799 C7U0TW 11747 Ki > 100000 nM T99799 C53FYO 11840 Ki > 100000 nM T99799 CKR3L9 12116 Ki > 100000 nM T99799 CU5KZ0 13005 Ki > 100000 nM T99799 CJ2GH1 13006 Ki > 100000 nM T99799 CG1LI5 14313 Ki > 100000 nM T99799 C4FW7E 18475 Ki > 100000 nM T99799 CTE5Z9 22006 IC50 = 14 nM T99799 C7S3JO 26257 Ki > 100000 nM T99799 C38JQX 31261 Ki > 100000 nM T99799 CN8A2G 38296 Ki > 100000 nM T99799 C7HE8W 38333 Ki > 100000 nM T99799 C0VK3I 39834 Ki > 100000 nM T99799 CVS6A8 40634 IC50 > 1000000 nM T99799 C8Z6TM 43402 Ki > 100000 nM T99799 CM94KL 47020 IC50 = 18000 nM T99799 CUNJ73 61209 Ki > 100000 nM T99799 C6U7FB 62539 Ki > 100000 nM T99799 C49ODY 65735 Ki = 610 nM T99799 C54XNY 68261 IC50 = 25100 nM T99799 C27NHT 69147 Ki > 100000 nM T99799 CN0ID1 69282 Ki > 100000 nM T99799 CW54JA 69288 Ki > 100000 nM T99799 C6BEN0 70945 Ki > 100000 nM T99799 C5KW4H 72311 IC50 = 10340 nM T99799 C2I7WP 74721 IC50 = 12000 nM T99799 CV8R4B 76561 Ki > 100000 nM T99799 CVJ78Y 79690 Ki > 100000 nM T99799 CAPG58 87502 Ki > 100000 nM T99799 C0EH3Z 88695 Ki > 100000 nM T99799 C70KGR 92036 Ki > 100000 nM T99799 C13IQL 93772 Ki > 100000 nM T99799 C8YU9Z 95415 Ki > 100000 nM T99799 CH91PI 95447 Ki > 100000 nM T99799 CAET12 101464 Ki = 90800 nM T99799 CR3E9L 103786 Ki > 100000 nM T99799 CG2VD5 120652 IC50 = 5248.07 nM T99799 CVB9H1 121587 IC50 > 50000 nM T99799 CVH8G6 122824 IC50 = 1600 nM T99799 C20LIY 136371 Ki > 100000 nM T99799 CTU83D 137777 Ki > 100000 nM T99799 CHAN02 138508 Ki > 100000 nM T99799 CYX5V0 142278 Ki > 100000 nM T99799 CF3I2J 156793 IC50 = 21770 nM T99799 C28RAT 165208 IC50 = 500 nM T99799 CIZE15 189688 IC50 > 100000 nM T99799 CX54PW 192442 IC50 = 3400 nM T99799 C5O8MF 197067 IC50 = 13680 nM T99799 C4VZL0 202767 IC50 > 1000000 nM T99799 C73HEY 203361 IC50 = 9800000 nM T99799 C1UW4K 204303 IC50 = 583000 nM T99799 CT8KV4 205772 IC50 = 52 nM T99799 C6W8MB 219592 Ki > 100000 nM T99799 COQ09W 219605 Ki > 100000 nM T99799 C25BHS 222475 Ki > 100000 nM T99799 CN35KE 222570 Ki > 100000 nM T99799 CP4W3S 229680 Ki > 100000 nM T99799 C0KV5M 236566 Ki > 100000 nM T99799 CE6U1D 237515 Ki > 100000 nM T99799 C92OSL 241331 Ki > 100000 nM T99799 C4N8IF 252525 IC50 > 30000 nM T99799 CHP1J7 262695 Ki > 100000 nM T99799 CDL3E1 262696 Ki > 100000 nM T99799 C6PU5E 270291 IC50 = 1570 nM T99799 CF62QN 275182 IC50 > 100000 nM T99799 C4HQ7V 284016 IC50 = 61010 nM T99799 CBR3Z7 302171 IC50 = 41300 nM T99799 CCSF19 303539 IC50 = 3026 nM T99799 C08WNV 317405 IC50 = 46770 nM T99799 CTMV50 321195 IC50 = 60000 nM T99799 CJ8RQ0 335358 IC50 = 1365 nM T99799 C5EI4Q 354120 Ki = 920 nM T99799 C5YJ7Z 359278 IC50 = 32 nM T99799 CHL04T 362574 IC50 = 800 nM T99799 CKS3U9 366710 Ki > 100000 nM T99799 C35JHV 385410 IC50 = 10320000 nM T99799 C5V0SH 386338 IC50 > 10000 nM T99799 C54EGJ 402658 IC50 = 26400 nM T99799 C9E5NG 402660 IC50 = 3300 nM T99799 CGKY63 402662 IC50 = 2300 nM T99799 CDCN80 402664 IC50 = 6700 nM T99799 C34VZP 402665 IC50 > 100000 nM T99799 C98AUK 402666 IC50 = 36000 nM T99799 C2SD4E 405589 IC50 > 50000 nM T99799 C7NU8P 409398 Ki = 17100 nM T99799 C5SFM6 412865 IC50 = 987 nM T99799 C18OIX 441064 IC50 > 100000 nM T99799 CLD6J9 441074 IC50 = 1230 nM T99799 CRN10Y 442113 IC50 = 4 nM T99799 CO9W4L 442854 IC50 = 35000 nM T99799 CE7GQ5 460616 IC50 = 1200 nM T99799 CQ3B5U 468188 IC50 = 5000 nM T99799 CU8GI1 468192 IC50 = 1100 nM T99799 CYMH94 471008 IC50 > 200000 nM T99799 CMO53J 475411 IC50 > 200000 nM T99799 C7U6FE 496015 IC50 = 2590 nM T99799 C0MI1O 513223 IC50 = 36000 nM T99799 CQ2F1V 513225 IC50 > 50000 nM T99799 CRI95J 513235 IC50 = 4200 nM T99799 CTWM69 586418 Ki > 100000 nM T99799 CH1E7N 590628 Ki > 100000 nM T99799 CCJQ96 599378 Ki > 100000 nM T99799 CL5E6W 607775 IC50 > 10000 nM T99799 CQ2M9X 638277 IC50 = 13000 nM T99799 CN71BS 641819 IC50 = 42000 nM T99799 C9MC2E 657348 IC50 = 16 nM T99799 C9CL3E 662730 IC50 = 6030 nM T99799 CVSQ83 662866 IC50 = 781 nM T99799 CXIK27 667496 IC50 = 3130 nM T99799 CK5V3P 667498 IC50 = 2490 nM T99799 CR1E5K 667801 IC50 = 25500 nM T99799 CJG47Q 704266 Ki = 190 nM T99799 C3DPV8 705751 Ki = 35000 nM T99799 CQP4B1 705773 Ki = 560 nM T99799 CFL0Y1 719823 IC50 = 49580 nM T99799 C9GU2E 744392 Ki = 23400 nM T99799 C50NVY 784043 IC50 = 3900 nM T99799 C4TAX6 784405 IC50 = 4000 nM T99799 C7PO1F 787366 IC50 = 7700 nM T99799 CO6AH8 806726 Ki = 9630 nM T99799 CB3GD4 818016 Ki = 4894000 nM T99799 CI8K6W 818170 IC50 = 56450 nM T99799 C29EOV 830741 IC50 = 9300 nM T99799 CMSC64 854531 IC50 > 10000 nM T99799 C5E3VW 866335 IC50 = 4920 nM T99799 CI54UD 866337 IC50 = 1090 nM T99799 C4BI6D 927411 IC50 > 50000 nM T99799 CA4D9I 931706 IC50 = 9820 nM T99799 CD3V9G 938070 IC50 = 61550 nM T99799 C84UPO 1018444 IC50 > 50000 nM T99799 C1YHE8 1208238 IC50 = 16600 nM T99799 CE7QJ6 1234089 IC50 = 51340 nM T99799 CYXQ78 1234090 IC50 = 37920 nM T99799 CED67Q 1237217 Ki = 1500 nM T99799 CC8JS7 1241150 IC50 = 42600 nM T99799 C3ZT7O 1320633 Ki = 6910 nM T99799 CM0I1K 1371037 Ki = 23000 nM T99799 CR37OY 1489313 IC50 = 250000 nM T99799 CIK9V0 1593398 IC50 = 83 nM T99799 CWTV42 1713189 Ki = 21000 nM T99799 C0EX9G 1755771 Ki > 100000 nM T99799 CB0ZP3 1812008 Ki > 100000 nM T99799 C9HL7Z 1816914 IC50 = 54090 nM T99799 CL8YK1 1889619 Ki = 90 nM T99799 C3FQD8 1906162 Ki > 100000 nM T99799 C3O6MN 1972026 Ki > 100000 nM T99799 C3X7MN 1991974 Ki = 20500 nM T99799 CI6ZU8 2133593 IC50 > 100000 nM T99799 CF37ZA 2147394 Ki > 100000 nM T99799 C0BEM3 2175773 IC50 > 50000 nM T99799 CJD8B3 2305233 Ki = 18100 nM T99799 CC5LI4 2326820 Ki = 2700 nM T99799 CN4U9J 2359994 IC50 = 5300 nM T99799 CC5J8U 2723754 IC50 = 23 nM T99799 CM6O4Z 2728673 IC50 = 57000 nM T99799 C68EBY 2728674 IC50 = 14000 nM T99799 C0OZQ2 2731126 Ki > 100000 nM T99799 CNKV06 2731127 Ki = 2390 nM T99799 CEM2C8 2731732 Ki > 100000 nM T99799 C2HOC5 2731733 Ki = 12300 nM T99799 CVC36I 2731902 Ki = 18900 nM T99799 CG62CN 2731904 Ki = 7400 nM T99799 CBEC45 2742082 IC50 > 30000 nM T99799 CN3KA4 2743222 IC50 < 10 nM T99799 C9R5LQ 2749125 Ki > 100000 nM T99799 C84DSN 2749126 Ki > 100000 nM T99799 CXU2J0 2755571 IC50 = 68000 nM T99799 C84VWR 2784639 Ki > 100000 nM T99799 CDCB42 2786143 Ki > 100000 nM T99799 C2RDM5 2886084 IC50 > 50000 nM T99799 CIK19R 2891624 IC50 = 443 nM T99799 CC8TY5 2915015 Ki = 7860 nM T99799 C6YQW9 2915964 Ki = 29100 nM T99799 CW9O2K 2930014 IC50 = 4.9 nM T99799 CRQ94D 2999234 IC50 > 100000 nM T99799 C1BM9V 3001811 IC50 > 200000 nM T99799 CC4OL6 3004425 Ki = 2150 nM T99799 CDR2K0 3012524 IC50 = 13880 nM T99799 C9QOY1 3029941 Ki = 510 nM T99799 CNYW30 3036637 IC50 = 529000 nM T99799 C04THC 3037884 IC50 = 1970 nM T99799 CZVE24 3041340 IC50 = 130000 nM T99799 C0JO2G 3055247 IC50 = 2400 nM T99799 CVN73X 3071771 IC50 = 25 nM T99799 CS5ET2 3071772 IC50 = 4100 nM T99799 CG09EQ 3071773 IC50 = 3100 nM T99799 CP2Y7N 3071774 IC50 = 3600 nM T99799 CZ6BA1 3071775 IC50 = 2900 nM T99799 C9M5PQ 3071776 IC50 = 1900 nM T99799 CI9VN7 3071777 IC50 = 1900 nM T99799 CC6W7T 3071778 IC50 = 1000 nM T99799 CIKF06 3071779 IC50 = 2700 nM T99799 CL2HU7 3071780 IC50 = 1300 nM T99799 CC9S8H 3072501 IC50 = 1800 nM T99799 CBLG95 3072502 IC50 = 3800 nM T99799 CS3L6G 3072503 IC50 = 3300 nM T99799 CIW2K3 3072504 IC50 = 2400 nM T99799 C2KN6J 3072505 IC50 = 3300 nM T99799 CEU74K 3072506 IC50 = 3800 nM T99799 CC56GR 3072507 IC50 = 1400 nM T99799 C4PCM1 3072508 IC50 = 4700 nM T99799 CHD8L0 3072509 IC50 = 6100 nM T99799 CU61MK 3072510 IC50 = 1300 nM T99799 CS1I6C 3072512 IC50 = 8400 nM T99799 CU20TQ 3072513 IC50 = 1600 nM T99799 C3KTC4 3072514 IC50 = 1100 nM T99799 C6QM9J 3072515 IC50 = 1800 nM T99799 CXLH39 3072518 IC50 = 5200 nM T99799 COW6E8 3075612 IC50 = 190 nM T99799 CU9Z2X 3083559 IC50 = 3000 nM T99799 CN5Z4H 3084319 IC50 = 2 nM T99799 CHEA42 3088389 IC50 = 4300 nM T99799 C1AM0S 3114312 Ki = 6710 nM T99799 C61RSW 3126152 Ki > 100000 nM T99799 CCP07Y 3264931 Ki > 100000 nM T99799 CB21VL 3321360 Ki > 100000 nM T99799 CZV6G2 3329233 Ki > 100000 nM T99799 C6NH9P 3469206 Ki > 100000 nM T99799 C3BT1N 3478673 IC50 = 45000 nM T99799 C10GCK 3527426 Ki > 100000 nM T99799 C3T1CV 3531512 Ki = 98900 nM T99799 CY6A2H 3706065 IC50 = 62000 nM T99799 CBZ13K 3722393 IC50 = 55800 nM T99799 C7V5YL 3748227 IC50 = 12200 nM T99799 CN5TX0 3756584 IC50 > 20000 nM T99799 CFV75H 3787603 IC50 = 4760 nM T99799 CV83OP 3796877 IC50 = 64800 nM T99799 C5UM2D 3821945 Ki > 100000 nM T99799 CU17BR 4088910 Ki > 100000 nM T99799 CR2X0V 4244497 Ki = 4690 nM T99799 CC1GF9 4338240 Ki > 100000 nM T99799 C8KV7I 4350924 Ki > 100000 nM T99799 C0V6QI 4369935 Ki > 100000 nM T99799 C42FGN 4384851 Ki > 100000 nM T99799 C01JRU 4416990 IC50 = 9100 nM T99799 CN9C3V 4513067 Ki > 100000 nM T99799 CAOH69 4789430 IC50 > 30000 nM T99799 CK9AT5 4792504 IC50 = 14000 nM T99799 CDV3O6 4846969 IC50 = 3000 nM T99799 C9MY1I 4885038 IC50 = 120 nM T99799 C5NJ3A 5004413 Ki > 100000 nM T99799 CNMY06 5038499 Ki > 100000 nM T99799 CL69XS 5127299 IC50 = 762 nM T99799 C7A0CD 5152006 IC50 = 2000 nM T99799 C0D3PO 5281671 IC50 = 1700 nM T99799 C5LGJ1 5282362 IC50 > 500000 nM T99799 C73SJW 5318015 IC50 > 100000 nM T99799 C5S6GW 5367146 IC50 = 105000 nM T99799 C32RHP 5367166 IC50 = 32000 nM T99799 C8HQN1 5376026 IC50 > 10000 nM T99799 CAC70Q 5377323 IC50 = 32000 nM T99799 CP1DZ2 5383464 IC50 = 27000 nM T99799 C25YUO 5458190 IC50 = 3170 nM T99799 C71CMO 5459840 IC50 = 506 ug.mL-1 T99799 CH6DT9 5481958 IC50 = 1700 nM T99799 CC6IV0 5481968 IC50 = 1700 nM T99799 CH8AJ6 5481969 IC50 = 1700 nM T99799 CMOI48 5481973 IC50 = 1700 nM T99799 CP69QB 5702326 IC50 > 5000 nM T99799 C81LVR 5702328 IC50 > 5000 nM T99799 CP46OW 5713121 IC50 = 1600 nM T99799 CGHW32 5747382 IC50 = 5100 nM T99799 C9L6KZ 5919802 IC50 = 31590 nM T99799 CYP0F4 6145899 IC50 = 119000 nM T99799 CR67NI 6333010 IC50 = 10 nM T99799 CK2MJ6 6333011 IC50 = 40 nM T99799 C8SZQ4 6410685 IC50 = 10000 nM T99799 C16EFR 6479925 IC50 = 100 nM T99799 CIL06S 6486743 IC50 = 18800 nM T99799 CNB34I 6540271 IC50 = 0.77 nM T99799 CW93TX 6610268 IC50 = 2140 nM T99799 C6EFT0 6712920 IC50 = 222 nM T99799 CSCO59 7580042 IC50 = 26070 nM T99799 C7BZ0N 7945979 IC50 > 5000 nM T99799 C9L0JT 9574517 IC50 = 240 nM T99799 CSY0F8 9574537 IC50 > 50000 nM T99799 CCLX43 9579448 IC50 = 2600 nM T99799 CK37WV 9579449 IC50 > 50000 nM T99799 C8XKM7 9794806 IC50 = 100 nM T99799 CU2XN7 9819233 IC50 = 1560 nM T99799 CFHP83 9822470 IC50 = 1570 nM T99799 CVDM07 9828345 IC50 = 257 nM T99799 CG6W8R 9839754 IC50 = 920 nM T99799 C7C0IP 9843814 Ki = 1400 nM T99799 CM0BX3 9850331 IC50 = 164 nM T99799 CKA8W7 9851127 IC50 = 194 nM T99799 C4VHS5 9859456 IC50 = 3100 nM T99799 CF05ZV 9864626 IC50 = 51 nM T99799 C2NLZ5 9886877 IC50 = 28100 nM T99799 CME5I4 9894056 IC50 = 26 nM T99799 C94UJV 9905831 IC50 = 1560 nM T99799 CE8M7Y 9928503 Ki = 20 nM T99799 CE69LQ 9952812 IC50 > 10000 nM T99799 CFW16Y 9958700 IC50 = 132 nM T99799 CYLG46 9959612 IC50 = 5.66 nM T99799 CC3G7N 9961034 IC50 = 3.3 nM T99799 CP3QN4 9976101 IC50 = 4800 nM T99799 C2WYT7 9976761 IC50 = 3900 nM T99799 CFH1O0 9992823 IC50 = 6.8 nM T99799 CI3D7M 10038341 IC50 = 59.4 nM T99799 CH0R1M 10038557 IC50 > 50000 nM T99799 C30ZHN 10040889 IC50 = 4300 nM T99799 CN0HU2 10044997 IC50 = 155000 nM T99799 CI2X0Z 10075220 IC50 = 0.6 nM T99799 CEKX28 10094001 IC50 > 50000 nM T99799 CWD41K 10097011 IC50 = 13.9 nM T99799 CTI26V 10098048 IC50 > 200000 nM T99799 CI70JE 10109540 IC50 > 50000 nM T99799 C68RJB 10110147 IC50 = 9000 nM T99799 CTQ95J 10110914 IC50 = 4200 nM T99799 CVWT04 10117403 IC50 = 13650 nM T99799 CSX92P 10126521 IC50 > 50000 nM T99799 C1B9MQ 10150601 IC50 > 50000 nM T99799 CA5J4V 10150622 IC50 > 50000 nM T99799 CO6I2N 10159339 IC50 = 890 nM T99799 CMJ4S6 10161755 IC50 = 31550 nM T99799 CV65OE 10179120 IC50 = 780 nM T99799 CQB9D0 10200831 IC50 = 26700 nM T99799 CD0P4U 10204915 IC50 = 22190 nM T99799 CS9E7Y 10205836 IC50 = 15670 nM T99799 C36DNM 10215997 IC50 > 50000 nM T99799 CP1HT3 10223679 IC50 = 250 nM T99799 CX4Y1T 10224148 IC50 = 15230 nM T99799 CY6I8F 10243365 Ki = 685200 nM T99799 CWZ5S0 10245631 IC50 = 516 nM T99799 CU6B5G 10255032 IC50 = 4840 nM T99799 C81ONP 10255275 IC50 = 18000 nM T99799 C8MAO5 10268794 Ki = 210 nM T99799 CD89EN 10272949 IC50 = 10790 nM T99799 C3GMK4 10277339 IC50 = 38400 nM T99799 CM19RC 10277340 IC50 = 57870 nM T99799 C7ZIP3 10277830 IC50 = 23210 nM T99799 CB2K1F 10287897 IC50 > 50000 nM T99799 C0TWQ3 10292083 IC50 = 6200 nM T99799 C08TOG 10299954 IC50 = 26830 nM T99799 C72VTB 10300579 IC50 = 78920 nM T99799 CV5B1A 10308583 IC50 > 50000 nM T99799 CJ0VN5 10310052 IC50 > 50000 nM T99799 C7NRO3 10317909 IC50 = 75000 nM T99799 CPRK30 10337156 IC50 = 23500 nM T99799 C4Z7DT 10337617 IC50 = 300000 nM T99799 CGZ5B9 10342292 IC50 = 1700 nM T99799 C1VFO0 10355816 IC50 > 2000 nM T99799 CRI5E2 10360601 IC50 = 1 nM T99799 C3H0MY 10372514 IC50 = 2238.72 nM T99799 CC5WG8 10416369 IC50 = 4.9 nM T99799 CB0VE3 10458051 IC50 = 31200 nM T99799 CI7C9Y 10464995 IC50 > 10000 nM T99799 CFN3I9 10472189 IC50 = 101910 nM T99799 CU21VN 10476544 IC50 > 50000 nM T99799 CHM50O 10481357 IC50 = 10.4 nM T99799 C7J2KT 10502606 IC50 = 776 nM T99799 CK5W8X 10505674 IC50 = 641 nM T99799 CGH7U6 10526350 IC50 = 85800 nM T99799 CWUY91 10539341 IC50 = 18900 nM T99799 C98RWG 10545891 IC50 = 21.8 nM T99799 CM3UP4 10550262 IC50 = 91200 nM T99799 CJ0N1R 10569957 IC50 = 1589.5 nM T99799 CIS15A 10573780 IC50 = 85.3 nM T99799 CYSD36 10593041 IC50 = 1430 nM T99799 C3XYI4 10597848 IC50 = 7086 nM T99799 CVD9A1 10610498 IC50 = 237 nM T99799 CTM40A 10615903 IC50 = 1745.5 nM T99799 C2LRS9 10622407 IC50 = 600 nM T99799 CV1PG0 10623652 IC50 = 85 nM T99799 CY93KL 10625415 IC50 = 53 nM T99799 CWE41Q 10655805 Ki > 100000 nM T99799 CZ59MX 10663695 IC50 = 396 nM T99799 CL95NU 10664401 IC50 = 730 nM T99799 CSIC19 10690207 IC50 = 78 nM T99799 CNR15Z 10713570 IC50 = 340 nM T99799 CG4Z8N 10721720 IC50 = 0.69 nM T99799 CL1BE8 10729509 IC50 = 42000 nM T99799 CRD47N 10730136 IC50 = 1120.5 nM T99799 CT68IS 10757271 IC50 = 952 nM T99799 C4O5KP 10763156 IC50 = 43800 nM T99799 CDAR18 10764956 IC50 = 8.1 nM T99799 C2AN5S 10774819 IC50 = 5900 nM T99799 CFHV29 10778312 IC50 = 197 nM T99799 C9PTG2 10785532 IC50 = 310 nM T99799 C4YS9A 10789991 IC50 = 156270 nM T99799 C9YLN1 10799366 IC50 = 12200 nM T99799 CKZ53Y 10825928 IC50 = 81000 nM T99799 CD0L7C 10848598 IC50 > 2000 nM T99799 C8G6BS 10850978 IC50 = 46 nM T99799 CGL0K9 10855014 IC50 = 2511.89 nM T99799 C8XSW2 10863593 Ki = 16200 nM T99799 CHF26C 10872974 IC50 = 270 nM T99799 CF28NJ 10879668 Ki > 100000 nM T99799 C3HZ6S 10894911 IC50 = 510 nM T99799 C1PZ2V 10896395 IC50 = 16.5 nM T99799 CH49NV 10899196 Ki > 100000 nM T99799 CP93JE 10902085 Ki > 100000 nM T99799 C95XSO 10905408 IC50 = 280 nM T99799 CU4W9S 10909176 IC50 = 758.58 nM T99799 CV35KR 10909236 IC50 = 2570.4 nM T99799 CSW4G1 10915203 IC50 = 815 nM T99799 C4M3ZI 10919451 IC50 = 8317.64 nM T99799 CR19FE 10927360 IC50 = 25 nM T99799 C3DSY6 10927599 IC50 = 42.6 nM T99799 CCS2Y7 10941381 IC50 = 7413.1 nM T99799 C0I9NT 10943454 IC50 > 10000 nM T99799 CZSC17 10958661 IC50 > 10000 nM T99799 C2Y5XC 10961666 IC50 = 3650 nM T99799 C2WRK0 10963725 IC50 = 165.96 nM T99799 CK72HO 10974737 IC50 = 165958.69 nM T99799 CJ7DR2 10985959 IC50 = 7585.78 nM T99799 CQ4ZC5 10996738 IC50 = 1659.59 nM T99799 C4NY9F 11006704 IC50 = 3.9 nM T99799 CD96QS 11007082 IC50 = 54954.09 nM T99799 C7NZY9 11009341 Ki > 100000 nM T99799 C9PTO8 11027124 IC50 = 53700 nM T99799 C0F1HL 11027759 IC50 = 2000 nM T99799 CN6WF9 11051398 IC50 = 83.18 nM T99799 CO30RK 11081720 IC50 = 310600 nM T99799 CPSM68 11104192 IC50 = 2630.27 nM T99799 CSYM37 11104646 IC50 = 2137.96 nM T99799 CF15NS 11113449 Ki = 3400 nM T99799 CJ0RG8 11113852 Ki = 26300 nM T99799 CUZ1H3 11114008 IC50 > 30000 nM T99799 C74KUO 11115691 IC50 = 6456.54 nM T99799 CJ2P6K 11121264 IC50 > 10000 nM T99799 CST19B 11124861 IC50 = 7.5 nM T99799 CKJ49N 11125225 IC50 = 5495.41 nM T99799 CKRZ24 11125922 IC50 = 1412.54 nM T99799 C1Q5OP 11136870 IC50 = 2398.83 nM T99799 C7FPU3 11146640 IC50 = 1071.52 nM T99799 CIP41D 11150497 IC50 = 410 nM T99799 C8FNC1 11156231 IC50 = 0.03 nM T99799 C9LFS7 11156598 IC50 = 0.1 nM T99799 C7JC9B 11167725 IC50 = 16 nM T99799 CGWM68 11168014 IC50 = 206 nM T99799 C8UTA5 11169647 IC50 = 63.7 nM T99799 CYL18X 11179973 IC50 = 70300 nM T99799 C9IV7T 11181553 IC50 = 1621.81 nM T99799 C4EU7X 11188905 IC50 = 1000 nM T99799 C6L0IS 11190153 IC50 = 329 nM T99799 CZ2GU4 11191030 IC50 = 79 nM T99799 C3D5SL 11191634 IC50 = 3.4 nM T99799 CBJV46 11192468 IC50 = 40200 nM T99799 CM54US 11192952 IC50 = 84400 nM T99799 CSJ1R4 11193161 IC50 = 330 nM T99799 CH30SU 11204324 IC50 = 81300 nM T99799 CE21OG 11204682 IC50 = 15488.17 nM T99799 C9EMG6 11209350 IC50 = 2000 nM T99799 CZPB69 11210161 IC50 = 200 nM T99799 CJI9N3 11216927 IC50 = 1096.48 nM T99799 C7X9ZC 11221007 Ki = 860 nM T99799 C4N9ZL 11221206 IC50 = 100 nM T99799 C1NI8D 11222968 IC50 > 10000 nM T99799 CY86GP 11226206 IC50 = 44300 nM T99799 CX6CF4 11232205 IC50 = 130 nM T99799 CEXP98 11233503 IC50 = 27 nM T99799 CT38EP 11235216 IC50 > 50000 nM T99799 C6TVW3 11238481 IC50 = 500 nM T99799 CSXF65 11238662 IC50 = 610 nM T99799 CV73WE 11239040 IC50 = 761000 nM T99799 C5FO1B 11243200 IC50 = 370 nM T99799 C6GHQ3 11244670 IC50 = 14000 nM T99799 CRL20G 11249115 IC50 = 2.9 nM T99799 C8GJD2 11249560 IC50 = 5.7 nM T99799 C6LH1M 11250361 IC50 = 130000 nM T99799 C81GLD 11257074 IC50 = 8.3 nM T99799 CKTJ19 11260293 IC50 > 30000 nM T99799 CPSO84 11261638 IC50 = 9000 nM T99799 CP6FX1 11268904 IC50 = 900 nM T99799 CEBK83 11272051 IC50 = 22.4 nM T99799 CC14OZ 11272989 IC50 = 155000 nM T99799 CAP59Z 11278342 IC50 = 50 nM T99799 CYRB74 11283475 IC50 = 11.7 nM T99799 C2CQH5 11283831 IC50 = 4650000 nM T99799 C1JKX2 11290299 IC50 = 100 nM T99799 CE79LQ 11290672 IC50 = 2165 nM T99799 CXV91C 11304331 IC50 > 50000 nM T99799 CKD79X 11304963 IC50 = 47.5 nM T99799 CBL8D9 11314048 IC50 = 4000 nM T99799 C2SQ3D 11314386 IC50 > 50000 nM T99799 CX9JQ2 11316712 IC50 = 12 nM T99799 CAJ8O0 11316986 IC50 = 1 nM T99799 CEKG13 11329992 IC50 = 57900 nM T99799 C9JV3E 11330142 Ki = 8.59 nM T99799 CNTY27 11336871 IC50 = 460 nM T99799 C7RJ4Z 11341331 IC50 = 5.6 nM T99799 CG91BA 11350292 IC50 > 50000 nM T99799 CM34HL 11352229 IC50 = 3.24 nM T99799 CAR45P 11359651 IC50 = 900 nM T99799 C59YIW 11359764 IC50 = 24400 nM T99799 CK49FX 11364765 IC50 = 600 nM T99799 CSE62M 11365562 IC50 = 136000 nM T99799 CQU73N 11376655 IC50 = 40 nM T99799 CI0CV9 11378169 IC50 = 660.69 nM T99799 CIAR80 11380022 IC50 = 6 nM T99799 CPB6X4 11381434 IC50 > 10000 nM T99799 CFS5X7 11382561 IC50 = 10.4 nM T99799 CSDY73 11385572 IC50 = 5.04 nM T99799 C61VUW 11392125 IC50 = 4 nM T99799 CPNA70 11393196 IC50 > 30000 nM T99799 CJAL17 11397926 IC50 = 77 nM T99799 CWB6K1 11404631 IC50 = 416 nM T99799 C8W9AR 11409935 IC50 = 11.7 nM T99799 CR7E9T 11420352 IC50 = 5500 nM T99799 CXLY31 11425531 IC50 = 24 nM T99799 CL9G3Y 11425872 IC50 = 200 nM T99799 C7T8KU 11432076 IC50 = 3.2 nM T99799 C5DML9 11432727 IC50 = 600 nM T99799 C83YSD 11434003 IC50 = 95499.26 nM T99799 CY72LB 11438752 IC50 > 30000 nM T99799 CL15TO 11445385 IC50 = 8490 nM T99799 C5TOG0 11445610 IC50 = 2190 nM T99799 CS7U9F 11455392 IC50 = 21.4 nM T99799 CY3EG9 11457400 IC50 = 1862.09 nM T99799 CKU29D 11461464 IC50 = 612 nM T99799 CAE18Q 11464843 IC50 = 11400000 nM T99799 C2N7YB 11465667 IC50 = 1.7 nM T99799 CA92CF 11465956 IC50 = 19 nM T99799 C9E6RY 11478767 IC50 = 1.7 nM T99799 C1KBO3 11478903 IC50 = 94600 nM T99799 C19ONS 11482774 IC50 = 2 nM T99799 C3WVS4 11489952 Ki = 0.74 nM T99799 CFQ27V 11490183 IC50 = 400 nM T99799 CSQZ71 11495096 IC50 = 12 nM T99799 C7OR8M 11504245 IC50 = 3 nM T99799 C94WCH 11509353 IC50 = 1.09 nM T99799 CVN51A 11514475 IC50 = 3 nM T99799 CA07BP 11530167 IC50 = 5100 nM T99799 CHLC49 11539744 IC50 = 0.68 nM T99799 C4CA7T 11550697 IC50 = 120 nM T99799 CY9MU1 11563410 IC50 = 25 nM T99799 CPHO51 11566532 IC50 = 15 nM T99799 C9XNM6 11573923 IC50 = 54 nM T99799 CWI4A2 11574168 IC50 = 23 nM T99799 C6P0EV 11576166 IC50 = 20000 nM T99799 C48YEL 11581590 IC50 > 50000 nM T99799 CH04PB 11588880 IC50 = 0.87 nM T99799 C3WQI0 11595988 IC50 > 50000 nM T99799 C2C4KA 11599119 IC50 = 35 nM T99799 CK2PB1 11603489 IC50 = 0.25 nM T99799 CLOD63 11606144 IC50 = 23 nM T99799 COAU76 11620371 IC50 = 6.8 nM T99799 CSDF87 11624531 IC50 = 13 nM T99799 CAF5O0 11625278 IC50 = 0.89 nM T99799 C2LD0Q 11631221 IC50 = 52000 nM T99799 CV5RH1 11631680 IC50 = 1180 nM T99799 CMH6K9 11632307 IC50 = 5100 nM T99799 CEY1C7 11645534 IC50 = 11400 nM T99799 CQX1I8 11647230 IC50 = 82400 nM T99799 CBGT09 11648619 IC50 = 12.6 nM T99799 CAE18N 11653182 IC50 = 72 nM T99799 CU1K8W 11666118 IC50 = 28 nM T99799 C67HTG 11667904 IC50 > 50000 nM T99799 C27AHE 11668852 IC50 > 50000 nM T99799 C8E6NF 11669798 IC50 = 9.5 nM T99799 C0AR9Z 11681391 IC50 = 36400 nM T99799 CI5MT9 11681880 IC50 = 40 nM T99799 C47LNU 11682017 IC50 > 50000 nM T99799 CC1ZN6 11694595 IC50 = 23 nM T99799 CR1IW0 11697764 IC50 = 3600 nM T99799 C5HYV7 11698149 IC50 = 2490 nM T99799 CL41DM 11698541 IC50 > 50000 nM T99799 CJ6UR7 11706508 IC50 = 7.8 nM T99799 C71EWN 11713155 IC50 = 1 nM T99799 C5FJ0D 11722860 IC50 = 897 nM T99799 C45PDY 11734220 IC50 = 4000 nM T99799 CBY03I 11739675 IC50 = 22 nM T99799 C1SDF0 11752376 IC50 = 8.58 nM T99799 C51RYW 11752643 IC50 = 32 nM T99799 CLMV71 11753218 Ki = 3.13 nM T99799 CQB14T 11763573 IC50 = 153000 nM T99799 C7MFV8 11763757 IC50 = 18620.87 nM T99799 C7OPQ0 11772375 IC50 = 300 nM T99799 CV84AY 11776726 IC50 = 2.4 nM T99799 CV4W8C 11784091 IC50 = 480 nM T99799 CZRE80 11786613 IC50 = 100 nM T99799 CG34JX 11792247 IC50 = 1473 nM T99799 CQ6YH2 11799236 IC50 = 513 nM T99799 CS23AV 11800047 IC50 = 1.36 nM T99799 CCQN45 11805526 Ki > 100000 nM T99799 C7WYG3 11810853 IC50 = 1600 nM T99799 CX97ZV 11814517 IC50 = 4073.8 nM T99799 CVS5N8 11854653 IC50 = 1.7 nM T99799 CCH27V 12013999 IC50 = 18900 nM T99799 CTM34I 12109666 IC50 = 224670 nM T99799 CJC3N0 12146686 IC50 > 30000 nM T99799 CKG7A0 12222796 Ki > 100000 nM T99799 CC3MQ9 12314224 IC50 = 56 nM T99799 CD1J7E 12851056 Ki = 24700 nM T99799 C5L0GN 12927905 IC50 = 541000 nM T99799 C1R4MF 12995052 IC50 = 230 nM T99799 C54QHI 13006034 IC50 = 250 nM T99799 C6XHS1 13006035 IC50 = 1820 nM T99799 CG7AZ9 13006036 IC50 = 165 nM T99799 CDP08C 13006037 IC50 = 170 nM T99799 C0AH2N 13006038 IC50 = 66 nM T99799 CIY8G4 13006039 IC50 = 798 nM T99799 CTX5Q6 13006040 IC50 = 490 nM T99799 CJ43VT 13006041 IC50 > 10000 nM T99799 CS7V4K 13006042 IC50 = 5020 nM T99799 CT5C2K 13006043 IC50 = 3290 nM T99799 CH46IX 13006044 IC50 = 1100 nM T99799 C3VSW6 13006045 IC50 = 650 nM T99799 CFE3W8 13006046 IC50 = 3890 nM T99799 CU0BN1 13006047 IC50 = 8530 nM T99799 CAJG53 13300537 IC50 = 840000 nM T99799 C0KSR2 13497076 IC50 = 150000 nM T99799 CEO81S 13552185 IC50 = 1400000 nM T99799 CL4MK3 13552226 IC50 = 120000 nM T99799 C4TA0V 13735450 IC50 > 5000 nM T99799 C8B5LO 13780062 Ki > 100000 nM T99799 C3YOX2 13827082 Ki > 100000 nM T99799 C4CR1L 13827083 Ki > 100000 nM T99799 CK08BO 13896866 IC50 > 500000 nM T99799 C0TRN9 13934286 IC50 > 200000 nM T99799 CU2M9R 14107712 IC50 = 2489 nM T99799 C4YBN3 14109375 IC50 > 200000 nM T99799 CJS4R6 14193572 IC50 = 10 nM T99799 CM6R4N 14193573 IC50 = 3 nM T99799 C39VGI 14193575 IC50 = 3 nM T99799 C6BP1S 14193577 IC50 = 2 nM T99799 C0PO5M 14349781 IC50 = 290 nM T99799 CJZ46W 14353465 IC50 = 3570 nM T99799 C7NE3Y 14372818 IC50 = 41 nM T99799 CQA53V 14537189 Ki = 1300 nM T99799 CX7AE6 14537192 Ki = 800 nM T99799 CD0F5X 14537193 Ki = 4600 nM T99799 CTB5H2 14539882 IC50 = 1700 nM T99799 CULX32 14553493 IC50 = 1670 nM T99799 CH27JR 14609844 IC50 = 7883 nM T99799 C93MXE 14735915 IC50 = 53000 nM T99799 CAH47C 14735925 IC50 = 34000 nM T99799 CMF7U1 14877070 IC50 = 140000 nM T99799 CK69GO 15005009 IC50 = 18000 nM T99799 C6V9HJ 15005010 IC50 = 1100 nM T99799 C1EQ0S 15043261 IC50 = 17990 nM T99799 C8PYV9 15043264 IC50 = 18200 nM T99799 CL2C7Y 15044210 Ki > 100000 nM T99799 CNJ2A9 15085436 IC50 = 71 nM T99799 CJ3E7T 15125273 IC50 = 690 nM T99799 CA13LZ 15125274 IC50 = 4230 nM T99799 C9WTF1 15125278 IC50 = 2070 nM T99799 CVJP83 15289585 IC50 > 1000000 nM T99799 CZ3WJ2 15490813 IC50 = 273 nM T99799 C1S6GM 15720175 IC50 = 17 nM T99799 CR2J0F 16094841 IC50 = 12.1 nM T99799 C34FJR 16094854 IC50 = 12.8 nM T99799 C8JM2I 16094855 IC50 = 7.13 nM T99799 CCL15D 16094856 IC50 = 0.969 nM T99799 COID78 16094857 IC50 = 0.293 nM T99799 CMT73Z 16094858 IC50 = 6.03 nM T99799 C3RN7X 16094859 IC50 = 0.226 nM T99799 CWI3K1 16094860 IC50 = 0.141 nM T99799 CG14KR 16094871 IC50 = 27.6 nM T99799 CKJ3F6 16094872 IC50 = 1.68 nM T99799 CD9S2E 16094873 IC50 = 0.523 nM T99799 C35HXC 16094875 IC50 = 24 nM T99799 CU8W5V 16094876 IC50 = 0.139 nM T99799 CMKY94 16114893 IC50 > 50000 nM T99799 C9E6AH 16114898 IC50 > 50000 nM T99799 C4RCO2 16115141 IC50 > 50000 nM T99799 C28IBN 16219608 IC50 = 420 nM T99799 C6GD9H 16235993 IC50 > 5000 nM T99799 CFX56U 16407549 IC50 = 270 nM T99799 CG5J7B 16584800 IC50 = 214410 nM T99799 C6K4AZ 16645662 Ki = 45400 nM T99799 C7MSU0 16653132 IC50 > 100000 nM T99799 C1JKF6 16664256 IC50 = 555500 nM T99799 CH9Y5B 17159064 IC50 = 3500 nM T99799 C5ZMI9 17159212 IC50 = 7200 nM T99799 CF6ZW1 17159244 IC50 = 11000 nM T99799 C80YMT 17159252 IC50 = 7800 nM T99799 CL2IW7 17422256 IC50 = 1360 nM T99799 CM9AH0 17602492 IC50 = 10300 nM T99799 C91BCT 17652420 Ki = 42500 nM T99799 C2OF8S 18471933 Ki > 100000 nM T99799 CFD89G 18870980 IC50 = 656850 nM T99799 C2QZ4O 18870983 IC50 = 11020 nM T99799 C39VUS 19760985 IC50 = 10420 nM T99799 CW0H1Y 20055993 IC50 > 200000 nM T99799 CU5Y8N 20208765 IC50 = 61659.5 nM T99799 C0Q9VM 20208772 IC50 = 13803.84 nM T99799 C45TLN 21204337 IC50 = 51000 nM T99799 C0ET8M 21362734 IC50 > 10000 nM T99799 C72BMS 21409569 IC50 = 22700 nM T99799 CQKH16 21592283 IC50 = 188360 nM T99799 CJKR07 21632954 IC50 > 200000 nM T99799 CEJ49C 21633084 IC50 > 200000 nM T99799 C2FBA3 21672659 IC50 > 30000 nM T99799 CX8W6N 21839636 IC50 = 63.3 nM T99799 CT3YN1 21839638 IC50 = 543 nM T99799 C5GZ1L 21839640 IC50 = 32.4 nM T99799 C8YO3H 21839642 IC50 = 109 nM T99799 CWR90B 21839649 IC50 = 89 nM T99799 CI29XS 22064898 IC50 > 100000 nM T99799 CYUW32 22181436 IC50 = 36800 nM T99799 C1DL8N 22210859 IC50 = 570 nM T99799 CYF5N8 22210860 IC50 = 27000 nM T99799 CYQB56 22210861 IC50 = 26000 nM T99799 C10ZWQ 22210862 IC50 = 3900 nM T99799 CH5YQ0 22210863 IC50 = 1800 nM T99799 CM3Y1I 22574246 Ki > 100000 nM T99799 C5IZQ8 23093594 IC50 = 1400 nM T99799 CHO5K2 23102336 Ki = 150 nM T99799 C7KCD5 23247894 IC50 > 200000 nM T99799 CZ0L4G 23277102 IC50 = 46000 nM T99799 CK15SO 23448959 IC50 = 38600 nM T99799 C13RZX 23624871 IC50 = 505 nM T99799 CZ7ET2 23634635 IC50 > 10000 nM T99799 CQ91XS 23634752 IC50 > 10000 nM T99799 CSK7Z4 23634753 IC50 > 10000 nM T99799 COZ1U3 23634754 IC50 > 10000 nM T99799 CIR09L 23634873 IC50 > 10000 nM T99799 CJMI97 23634874 IC50 = 375 nM T99799 CO5D8M 23634876 IC50 = 1450 nM T99799 CNFK89 23635382 IC50 > 10000 nM T99799 C0LA7S 23635383 IC50 > 10000 nM T99799 C15ASX 23635398 IC50 > 50000 nM T99799 C9F1MQ 23635399 IC50 > 50000 nM T99799 CXIA45 23635400 IC50 > 50000 nM T99799 CQ0H4M 23635401 IC50 > 50000 nM T99799 CZ5R6B 23635511 IC50 > 50000 nM T99799 C5S2QB 23635512 IC50 > 50000 nM T99799 C4B8MX 23635513 IC50 > 50000 nM T99799 CWD7J8 23635514 IC50 > 50000 nM T99799 C0ASM1 23635515 IC50 > 50000 nM T99799 CKP70J 23635516 IC50 > 50000 nM T99799 CM0X3T 23635632 IC50 > 50000 nM T99799 C0VL9W 23635633 IC50 > 50000 nM T99799 CJ73KM 23635634 IC50 > 50000 nM T99799 CWI26H 23635635 IC50 > 50000 nM T99799 CP6J2G 23635636 IC50 > 50000 nM T99799 C4GA2J 23635637 IC50 > 50000 nM T99799 CTJ96S 23635746 IC50 > 10000 nM T99799 C1P7GL 23635748 IC50 > 10000 nM T99799 CV8QU5 23635749 IC50 > 10000 nM T99799 CT46CR 23635766 IC50 = 19000 nM T99799 CVJ6C0 23635767 IC50 > 50000 nM T99799 CU61DC 23635768 IC50 > 50000 nM T99799 C74DZC 23635875 IC50 = 1535 nM T99799 CGJ6U3 23635876 IC50 = 380 nM T99799 CF91IH 23635891 IC50 > 50000 nM T99799 CT67MK 23635892 IC50 > 50000 nM T99799 CKM0C8 23635893 IC50 > 50000 nM T99799 CC1PX4 23635894 IC50 > 50000 nM T99799 C0XQ8E 23635895 IC50 = 8200 nM T99799 CCPS26 23635896 IC50 > 50000 nM T99799 C4UY7R 23636019 IC50 > 50000 nM T99799 CHTN58 23636020 IC50 > 50000 nM T99799 CPV52Y 23636021 IC50 > 50000 nM T99799 CD71KA 23636022 IC50 > 50000 nM T99799 C6QA3I 23636023 IC50 > 50000 nM T99799 CQ4U9X 23636024 IC50 > 50000 nM T99799 C93CLQ 23644605 IC50 = 3.8 nM T99799 CMH24N 23644647 IC50 = 5.55 nM T99799 CQ49JO 23644649 IC50 = 4.74 nM T99799 C4HV8T 23644653 IC50 = 7.8 nM T99799 C01OPD 23644658 IC50 = 4 nM T99799 CSQ9L7 23644774 IC50 = 328 nM T99799 C3AS4O 23644775 IC50 = 165 nM T99799 C2V8TA 23644776 IC50 = 45 nM T99799 C5W0NY 23644777 IC50 = 312 nM T99799 C8YQA2 23644778 IC50 = 93 nM T99799 CPO4L8 23644779 IC50 = 59 nM T99799 CSU1T2 23644780 IC50 = 23 nM T99799 C38QZE 23644781 IC50 = 3.3 nM T99799 CZH24F 23644782 IC50 = 2.6 nM T99799 CM39BI 23645223 IC50 = 1.48 nM T99799 CW8F0V 23645224 IC50 = 2580 nM T99799 CTW9J8 23645267 IC50 = 7.69 nM T99799 CRB3O6 23645269 IC50 = 6.7 nM T99799 CB8H9A 23645271 IC50 = 14 nM T99799 C34ZIH 23645273 IC50 = 7.38 nM T99799 CK2NJ4 23645289 IC50 = 1560 nM T99799 C3RP5S 23648183 IC50 = 7407 nM T99799 CQ9VY0 23648184 IC50 > 10000 nM T99799 CC0S5M 23653045 IC50 = 6401 nM T99799 CG61EZ 23765385 IC50 = 15200 nM T99799 CR8CW5 24202660 IC50 > 50000 nM T99799 CANS31 24749809 IC50 = 11.3 nM T99799 C4Z2EB 24749810 IC50 = 35.1 nM T99799 C4FVB7 24749811 IC50 = 5.44 nM T99799 CO9D4U 24799948 IC50 = 5.5 nM T99799 C6LV5R 24799949 IC50 = 36.5 nM T99799 C8JPO2 24800125 IC50 = 28 nM T99799 C64FMN 24800126 IC50 = 5.2 nM T99799 C8GKX5 24800127 IC50 = 21.7 nM T99799 C6DSC8 24800128 IC50 = 9.9 nM T99799 CW7LB1 24800129 IC50 = 15.3 nM T99799 CZ14LB 24800130 IC50 = 13.5 nM T99799 C59BPF 24800294 IC50 = 12.1 nM T99799 C07CZO 24800295 IC50 = 15.1 nM T99799 C5H3EC 24800296 IC50 = 5.5 nM T99799 C0QLV7 24800297 IC50 = 13.8 nM T99799 CAO8P0 24800298 IC50 = 10.8 nM T99799 CARE83 24800299 IC50 = 41 nM T99799 CZ0GN5 24800469 IC50 = 7.3 nM T99799 CQNB75 24825630 Ki > 100000 nM T99799 CF6W3Z 24833568 IC50 = 6820 nM T99799 C82UXG 24841476 Ki = 2450 nM T99799 C08HVP 24841478 Ki = 2400 nM T99799 CY21RE 24841480 Ki = 650 nM T99799 CVZ3G8 24845717 IC50 = 4 nM T99799 CMF3P2 24845873 IC50 = 34000 nM T99799 CR6M2L 24863097 Ki = 0.819 nM T99799 CBP1Y5 24865177 IC50 = 280 nM T99799 COR9K5 24865178 IC50 = 1830 nM T99799 CIY6F4 24865179 IC50 = 38100 nM T99799 CKB7T5 24865359 IC50 = 40900 nM T99799 CS1VB7 24865360 IC50 = 1820 nM T99799 C50JUL 24865361 IC50 = 21700 nM T99799 CH0WZ8 24865362 IC50 = 89100 nM T99799 C9W8TE 24865363 IC50 = 74100 nM T99799 C2CX0D 24879253 Ki = 0.779 nM T99799 CO3D6F 24879256 Ki = 1.187 nM T99799 CE7RA8 24879313 Ki = 0.924 nM T99799 COVB34 24879315 Ki = 13.86 nM T99799 CX60OH 24879317 Ki = 0.27 nM T99799 CW49DK 24879319 Ki = 0.725 nM T99799 C3DGL7 24879377 Ki = 0.435 nM T99799 CQM5Y4 24879379 Ki = 4.191 nM T99799 CA6WB0 24879381 Ki = 3.223 nM T99799 CRWB78 24879383 Ki = 1.872 nM T99799 C3GTP2 24879451 Ki = 5.04 nM T99799 CDI31X 24879453 Ki = 7.29 nM T99799 C51PQF 24881876 IC50 = 12.3 nM T99799 CLM2P5 24881945 IC50 = 8.06 nM T99799 CDI95B 24881949 IC50 = 7.25 nM T99799 CM5NY1 24905533 Ki = 260000 nM T99799 CBM4Q0 24905591 Ki = 3200 nM T99799 C6ZWN0 24905654 Ki = 1910 nM T99799 CW81VH 24905655 Ki = 120 nM T99799 CABV24 24936088 Ki = 19500 nM T99799 CO1ID8 24949376 IC50 = 296 nM T99799 C5VL9C 24949523 IC50 = 211 nM T99799 C2UZ4A 24949524 IC50 = 189 nM T99799 C3OV2G 24949525 IC50 = 137 nM T99799 CDY49T 25016412 IC50 = 4000 nM T99799 CVQY09 25016666 IC50 = 800 nM T99799 C2OD8R 25022724 IC50 = 4650 nM T99799 CAVC47 25033601 IC50 = 400 nM T99799 CML5I0 25053470 IC50 = 49980 nM T99799 CEM9A4 25053473 IC50 = 5890 nM T99799 CCR8V4 25053476 IC50 = 1720 nM T99799 C5XJH0 25053537 IC50 = 4590 nM T99799 C9WL5U 25053538 IC50 = 7540 nM T99799 C18HXS 25129144 IC50 = 28 nM T99799 CP91JC 25129145 IC50 = 32 nM T99799 CA2P7V 25129146 IC50 = 12 nM T99799 CD5Z2O 25129487 IC50 = 137 nM T99799 CHN93D 25145301 IC50 = 14400 nM T99799 C3P4KA 25149263 IC50 = 2090 nM T99799 CX50VY 25149264 IC50 = 293 nM T99799 CU45TK 25149265 IC50 = 1910 nM T99799 CU7EV3 25149453 IC50 = 10700 nM T99799 CB9Q1Y 25149538 IC50 = 1040 nM T99799 CEF4M1 25150256 IC50 = 30800 nM T99799 CES10Z 25150257 IC50 = 25300 nM T99799 CW5Y9S 25150356 IC50 = 10300 nM T99799 C6KSF0 25150451 IC50 = 95.8 nM T99799 CEL09B 25150452 IC50 = 876 nM T99799 CKW2Z0 25150453 IC50 = 3000 nM T99799 CB7K2G 25150454 IC50 = 416 nM T99799 CSLH31 25204947 IC50 = 334 nM T99799 C9NG2M 25205011 IC50 = 7322 nM T99799 C0TWB6 25211256 IC50 = 10000 nM T99799 CRKA79 25221268 IC50 = 116000 nM T99799 C6R3VH 25396473 Ki = 2.71 nM T99799 CKJZ59 25396479 Ki = 27.05 nM T99799 C2WPI3 27666802 IC50 = 1320 nM T99799 CL89DY 35793912 IC50 = 15300 nM T99799 CKJ82C 38864639 IC50 > 100000 nM T99799 CH4UY3 41474021 IC50 > 100000 nM T99799 CZ6KB8 41527552 IC50 = 3930 nM T99799 CJ06DE 42597801 IC50 = 60700 nM T99799 CJX2O8 42598036 IC50 = 88800 nM T99799 CX4H1M 42598039 IC50 > 100000 nM T99799 C7GO1F 42598040 IC50 = 16200 nM T99799 CE6Y3Z 42598041 IC50 = 125000 nM T99799 C0X7NH 42598042 IC50 = 71500 nM T99799 CNGR23 42598273 IC50 = 172000 nM T99799 C8K3WA 42598274 IC50 = 44000 nM T99799 CF75TP 42598275 IC50 > 100000 nM T99799 CXZ19Y 42598510 IC50 = 33200 nM T99799 CBOI16 42598737 IC50 > 10000 nM T99799 C5ROV0 42603833 IC50 = 1290 nM T99799 C2UN9H 42618134 IC50 > 100000 nM T99799 CH6X2V 42618135 IC50 > 100000 nM T99799 CCAU57 42618136 IC50 > 100000 nM T99799 C0EO3S 42618137 IC50 > 100000 nM T99799 CH21YS 42618138 IC50 > 100000 nM T99799 C2D4GJ 42637909 IC50 > 100000 nM T99799 CE4Q1Z 42637910 IC50 = 11000 nM T99799 C1E5GI 43824597 IC50 > 30000 nM T99799 C7YR8O 44224102 IC50 = 223 nM T99799 CMQ73T 44241603 IC50 = 3640 nM T99799 CNME62 44247959 IC50 = 290 nM T99799 CN80WP 44269395 IC50 = 4270 nM T99799 C2CZM3 44287477 IC50 = 910 nM T99799 CRL89F 44288141 IC50 = 920 nM T99799 C0QZG6 44288635 IC50 = 31 nM T99799 CZ9CM8 44289029 IC50 = 27 nM T99799 CWI3J4 44298002 IC50 = 1790 nM T99799 C5IS3D 44314031 IC50 = 11000 nM T99799 C4PH1U 44316259 IC50 = 216000 nM T99799 C9Y8WR 44316260 IC50 = 790000 nM T99799 C4GXD1 44316606 IC50 = 960000 nM T99799 CO6FT7 44328449 IC50 = 28000 nM T99799 C8KHN0 44328476 IC50 = 350 nM T99799 CIL4P7 44328516 IC50 = 3300 nM T99799 CK2UH8 44328517 IC50 = 2000 nM T99799 CLDZ15 44328518 IC50 = 48000 nM T99799 CD7VA3 44328527 IC50 > 50000 nM T99799 CY76FG 44328582 IC50 = 22000 nM T99799 CLB58A 44328594 IC50 > 50000 nM T99799 CY17DP 44328595 IC50 > 50000 nM T99799 CAEI14 44328600 IC50 = 2800 nM T99799 CJ10IH 44328655 IC50 = 4400 nM T99799 C27RNL 44328656 IC50 = 8800 nM T99799 CO75SD 44328657 IC50 = 2700 nM T99799 CU0VD3 44328667 IC50 = 3400 nM T99799 CYH27G 44328671 IC50 = 1000 nM T99799 CT0V8E 44328705 IC50 = 5600 nM T99799 C3T7KM 44328731 IC50 = 4400 nM T99799 CH5T7O 44328735 IC50 > 50000 nM T99799 CQ91KO 44328757 IC50 = 40000 nM T99799 C0BVX1 44328784 IC50 = 1200 nM T99799 CB9D2W 44328828 IC50 = 13000 nM T99799 CNU4R7 44328837 IC50 = 3900 nM T99799 CR97EP 44328842 IC50 = 250 nM T99799 CPE7B1 44328853 IC50 > 50000 nM T99799 CJ8Y0L 44328854 IC50 = 410 nM T99799 CR43YN 44338975 IC50 = 115 nM T99799 CUVK87 44339289 IC50 = 512 nM T99799 CT72FC 44339352 IC50 = 449 nM T99799 C0XI2G 44344490 IC50 = 88000 nM T99799 CZM80K 44344737 IC50 = 10300 nM T99799 CT1Q3S 44347198 IC50 = 50 nM T99799 CPXK27 44347214 IC50 = 2900 nM T99799 CNY9B1 44347584 IC50 = 1560 nM T99799 CVL5Y1 44347602 IC50 = 1950 nM T99799 CXD43V 44358068 IC50 = 2100 nM T99799 C05RBY 44358110 Ki = 1600 nM T99799 C3OPV1 44358179 Ki = 7500 nM T99799 CC79ZF 44361495 IC50 = 963 nM T99799 CK6QX1 44361516 IC50 = 331 nM T99799 CGHX23 44361622 IC50 = 32.6 nM T99799 C3OHM0 44361641 IC50 = 194 nM T99799 CF4GR3 44361719 IC50 = 1210 nM T99799 C0SZQ9 44362025 IC50 = 148 nM T99799 CF3H1M 44362158 IC50 = 63 nM T99799 C4L1OJ 44364861 Ki = 3250 nM T99799 CJKS01 44364863 Ki = 8600 nM T99799 CB6S7Y 44364908 IC50 = 2300 nM T99799 C39BIX 44385143 IC50 = 870.96 nM T99799 C3YO4B 44385678 IC50 = 270 nM T99799 C7Y0RT 44385890 IC50 > 2000 nM T99799 CP5FZ7 44386430 IC50 = 1410 nM T99799 CO6E7R 44386491 IC50 > 2000 nM T99799 CA5MZ0 44386492 IC50 > 2000 nM T99799 C5LXT8 44386641 IC50 > 2000 nM T99799 C61PJT 44386933 IC50 = 350 nM T99799 C9V2XH 44387832 IC50 = 3.9 nM T99799 C57WPN 44388351 IC50 = 17 nM T99799 CW09ZP 44391786 IC50 > 200000 nM T99799 CPZ3Y1 44391798 IC50 > 200000 nM T99799 C8XH3P 44391811 IC50 > 200000 nM T99799 C46ESP 44391828 IC50 > 200000 nM T99799 C56SXM 44391858 IC50 > 500000 nM T99799 CNBR80 44398165 IC50 = 24.5 nM T99799 C5P4KS 44398279 IC50 = 1.26 nM T99799 CX01VE 44398294 IC50 = 44.41 nM T99799 CN6PS1 44398377 IC50 = 10.5 nM T99799 C1M3ZD 44398397 IC50 = 209 nM T99799 C2B5HS 44398438 IC50 = 30.3 nM T99799 C7IRF1 44398566 IC50 = 74800 nM T99799 CMF05N 44409456 IC50 = 2 nM T99799 CJ35GS 44409574 IC50 = 4 nM T99799 C9ZHL5 44412131 Ki = 20.8 nM T99799 CQ12BX 44412132 Ki = 30.8 nM T99799 CHO3A1 44412135 Ki = 19.5 nM T99799 C4KN6X 44412186 IC50 = 15.8 nM T99799 CF0XV9 44417532 IC50 = 3980 nM T99799 C5MBE6 44417537 IC50 = 8490 nM T99799 C98SME 44417548 IC50 > 10000 nM T99799 CV7XP1 44417560 IC50 = 601 nM T99799 CVSZ87 44417568 IC50 > 10000 nM T99799 C0SR2L 44417569 IC50 = 9220 nM T99799 C0JYP1 44418744 IC50 = 1.38 nM T99799 CG41JA 44419699 IC50 > 10000 nM T99799 CY8RQ9 44419966 IC50 > 10000 nM T99799 CXZ52T 44419971 IC50 > 10000 nM T99799 CBD4I8 44421020 IC50 = 2300 nM T99799 C7SN0Z 44421297 IC50 = 11748.98 nM T99799 C9I7EY 44421298 IC50 = 2238.72 nM T99799 CD3SJ4 44421300 IC50 = 6456.54 nM T99799 CJ47UB 44421301 IC50 = 3630.78 nM T99799 C8GY2A 44421302 IC50 = 3388.44 nM T99799 CC64OM 44421303 IC50 = 1862.09 nM T99799 CV7RQ4 44421304 IC50 = 1819.7 nM T99799 CQ8V9A 44421305 IC50 = 1698.24 nM T99799 C6MFY8 44421520 IC50 = 136 nM T99799 CB9AO4 44421521 IC50 = 60 nM T99799 C03AEP 44421525 IC50 = 59 nM T99799 CM6IW2 44421529 IC50 = 9.6 nM T99799 CKNV25 44421531 IC50 = 54 nM T99799 CV46OY 44421933 IC50 = 63800 nM T99799 CHQ74U 44421934 IC50 = 127000 nM T99799 CM2PQ9 44421939 IC50 = 29500 nM T99799 CPM30V 44421940 IC50 = 14000 nM T99799 CX7T8G 44421945 IC50 = 2010 nM T99799 CGN9K0 44421946 IC50 = 1270 nM T99799 CR4K2Y 44421950 IC50 = 1000 nM T99799 CF0SC4 44421951 IC50 = 320 nM T99799 CH9WV0 44421967 IC50 = 46100 nM T99799 CQ6ZY2 44421972 IC50 = 3080 nM T99799 C4AF3S 44421973 IC50 = 1910 nM T99799 CO97PS 44421976 IC50 = 930 nM T99799 C1SK6X 44421982 IC50 = 1850 nM T99799 C9FZP5 44421986 IC50 = 2110 nM T99799 CTD13B 44421991 IC50 = 269000 nM T99799 CCB15K 44423472 IC50 = 29000 nM T99799 CEQ6U7 44423479 IC50 = 100 nM T99799 CO9LC6 44427467 IC50 = 279000 nM T99799 CM6GB7 44427468 IC50 > 0.00001 nM T99799 CEVO25 44427469 IC50 = 570000 nM T99799 CJ64GU 44427470 IC50 = 136000 nM T99799 CZ83QC 44427471 IC50 = 1300000 nM T99799 CPM03B 44427472 IC50 > 0.00001 nM T99799 CCJH84 44427473 IC50 > 0.00001 nM T99799 CN5CJ2 44427474 IC50 > 0.00001 nM T99799 CHQ62N 44427475 IC50 > 0.00001 nM T99799 C6WDH3 44427476 IC50 > 0.00001 nM T99799 CZTU76 44427477 IC50 > 0.00001 nM T99799 CO1NJ5 44427478 IC50 = 52900 nM T99799 CQ5G6X 44427479 IC50 > 0.00001 nM T99799 C4M7RQ 44427480 IC50 > 0.00001 nM T99799 CLS78U 44427481 IC50 = 35100 nM T99799 C5O1RW 44427482 IC50 > 0.00001 nM T99799 C0AM6W 44427483 IC50 > 0.00001 nM T99799 CE09QX 44427485 IC50 > 0.00001 nM T99799 CFMN40 44427486 IC50 > 0.00001 nM T99799 CS3AX5 44427487 IC50 > 0.00001 nM T99799 C9XM2E 44427488 IC50 > 0.00001 nM T99799 C0WMB1 44427489 IC50 > 0.00001 nM T99799 CPM76T 44427490 IC50 > 0.00001 nM T99799 CQ87RG 44427491 IC50 = 88900 nM T99799 CT38CX 44427492 IC50 > 0.00001 nM T99799 CSO3M0 44427493 IC50 = 43800 nM T99799 CDE8A1 44428745 IC50 = 10471.29 nM T99799 C0C2DX 44428836 Ki > 100000 nM T99799 CZS9U1 44428842 Ki > 100000 nM T99799 CWR3Y1 44428843 Ki > 100000 nM T99799 CUT0H7 44428844 Ki > 100000 nM T99799 C0NHI2 44435121 IC50 > 50000 nM T99799 CZ3RM2 44435219 Ki = 28 nM T99799 CIW9A7 44435348 IC50 > 1000 nM T99799 CV5Q1B 44435447 IC50 > 10000 nM T99799 CG7QK6 44435498 IC50 > 10000 nM T99799 CKP0Q3 44435526 IC50 = 1440 nM T99799 C83BXH 44435798 Ki > 100000 nM T99799 CF9SH8 44446101 Ki = 20400 nM T99799 C5K6XG 44446102 Ki = 754200 nM T99799 C7IH4Y 44446104 Ki = 161300 nM T99799 CE7M5J 44446106 Ki = 273800 nM T99799 CIQ4O9 44446113 Ki = 174500 nM T99799 CJ41TE 44550606 IC50 = 3000 nM T99799 CTYA64 44550607 IC50 = 730 nM T99799 CP0O8Q 44550608 IC50 = 70 nM T99799 CPWV46 44550725 IC50 = 1750 nM T99799 CQV8G2 44550726 IC50 = 1800 nM T99799 CNP4T9 44550727 IC50 = 850 nM T99799 CPT1O4 44550728 IC50 = 330 nM T99799 CLFZ14 44550729 IC50 = 830 nM T99799 CLVX32 44550849 IC50 = 350 nM T99799 CG1NK0 44562321 IC50 = 10000 nM T99799 CRA0U2 44562335 IC50 = 22060 nM T99799 CVA67X 44568347 Ki = 740 nM T99799 C0G8AC 44568806 IC50 = 2800 nM T99799 CJDG06 44568807 IC50 = 73 nM T99799 C0G3SJ 44580530 Ki = 1198 nM T99799 C1AO5C 44580576 Ki = 252 nM T99799 C9G1VW 44580577 Ki = 580 nM T99799 C5G2VP 44580578 Ki = 708 nM T99799 CP4FT6 44580579 Ki = 251 nM T99799 C6PLC4 44580639 Ki = 1764 nM T99799 CB1ZL8 44580640 Ki = 443 nM T99799 CQ6U4X 44580641 Ki = 173 nM T99799 CL73ZJ 44580642 Ki = 1.87 nM T99799 CK4M5S 44580643 Ki = 1.33 nM T99799 C8N4ZQ 44580644 Ki = 12.63 nM T99799 CMR90Y 44580645 Ki = 25.15 nM T99799 CWHP70 44580646 Ki = 1.77 nM T99799 CGJ3O4 44586009 IC50 = 196 nM T99799 CRJC18 44587246 IC50 = 1600 nM T99799 CM27UT 44587247 IC50 = 600 nM T99799 CKZJ17 44587345 IC50 = 29400 nM T99799 CP4G7M 44587346 IC50 = 76600 nM T99799 C37PVZ 44587494 IC50 = 4700 nM T99799 CMP67W 44587524 IC50 = 75200 nM T99799 C2CV9M 44587525 IC50 = 34400 nM T99799 CGK71P 44587544 IC50 = 3970 nM T99799 CI2L4T 44587564 IC50 = 19700 nM T99799 CIF0E9 44587921 IC50 = 142100 nM T99799 C7MW1Z 44589810 IC50 = 36800 nM T99799 CL1PQ6 44604353 IC50 > 30000 nM T99799 C34RFE 44604423 IC50 > 30000 nM T99799 C6K8GE 45049498 IC50 = 40000 nM T99799 CTBO39 45130737 IC50 = 345000 nM T99799 COF81U 45164786 IC50 = 2150 nM T99799 C5U6GX 45214445 IC50 = 21 nM T99799 CJP71Z 45261769 IC50 = 22.1 nM T99799 C2MN6D 45261778 IC50 = 24.5 nM T99799 CTYU71 45261781 IC50 = 31.6 nM T99799 CY6GX3 45261793 IC50 = 529 nM T99799 CZ16LQ 45261805 IC50 = 205 nM T99799 C67KQI 45261809 IC50 = 48.3 nM T99799 CW09OL 45261830 IC50 = 16.5 nM T99799 CY17RU 45263524 IC50 = 11600 nM T99799 CGE36P 45265144 IC50 = 34.1 nM T99799 CH6SJ9 45265175 IC50 = 25.2 nM T99799 CHA28P 45265179 IC50 = 24.8 nM T99799 COW2D8 45266157 IC50 = 660 nM T99799 CHE19F 45266158 IC50 > 10000 nM T99799 CNJ5W8 45266159 IC50 > 10000 nM T99799 C1LOR7 45266221 IC50 = 1700 nM T99799 CO9LU8 45266222 IC50 = 5200 nM T99799 CT01NJ 45267086 IC50 = 21100 nM T99799 CP5BH2 45269663 IC50 = 98100 nM T99799 C4HD1L 45269664 IC50 = 25000 nM T99799 CO4K0N 45269909 IC50 > 10000 nM T99799 CG92KC 45270503 IC50 = 175800 nM T99799 C3GF6X 45481996 IC50 = 2350 nM T99799 CQ4XH0 45481997 IC50 = 824 nM T99799 CJW20I 45482019 IC50 = 342 nM T99799 CAM26F 45482095 IC50 = 148000 nM T99799 C34LEX 45482096 IC50 = 31000 nM T99799 CK4Z8S 45482098 IC50 = 50000 nM T99799 C2CNM7 45482099 IC50 = 16100 nM T99799 CHMS72 45482100 IC50 = 133000 nM T99799 CYSP25 45482101 IC50 = 4200 nM T99799 CPT8J4 45482102 IC50 = 13400 nM T99799 C8ETA6 45482104 IC50 = 760 nM T99799 CDPT02 45482105 IC50 = 22000 nM T99799 CRO52I 45482106 IC50 = 140 nM T99799 CKE2N4 45487235 IC50 = 117 nM T99799 CG5W3E 45487242 IC50 = 0.15 nM T99799 C2VC7M 45487244 IC50 = 16 nM T99799 CF8M9K 45487246 IC50 = 323 nM T99799 CBTU95 45487247 IC50 = 18 nM T99799 C6B1IN 45487248 IC50 = 27 nM T99799 CG1ZJ8 45487252 IC50 = 86 nM T99799 CSQ78Z 45487253 IC50 = 297 nM T99799 C2SH7T 45487255 IC50 = 39 nM T99799 CLS2D9 45487263 IC50 = 32 nM T99799 CMJB89 45487264 IC50 = 9.6 nM T99799 CJ20LD 45487265 IC50 = 6.4 nM T99799 CBHD59 45487269 IC50 = 2609 nM T99799 C7S8KN 45487275 IC50 = 1057 nM T99799 CQFC83 45488333 IC50 > 5000 nM T99799 CW68OR 45490978 IC50 = 9570 nM T99799 C5IOS9 45490990 IC50 = 37400 nM T99799 C91TIQ 46204460 IC50 = 450300 nM T99799 CIG1O6 46211767 IC50 = 16210 nM T99799 CC64KH 46227076 IC50 = 19 nM T99799 C1MSE9 46228657 IC50 = 144000 nM T99799 C31MLQ 46228658 IC50 = 21100 nM T99799 CT9CI3 46228685 IC50 = 7930 nM T99799 CIK7S8 46228686 IC50 = 98100 nM T99799 C2V4QP 46228687 IC50 = 29900 nM T99799 CC85MY 46228688 IC50 = 22500 nM T99799 CE86KJ 46228721 IC50 = 11400 nM T99799 C7CY5S 46228722 IC50 = 22900 nM T99799 C7W8OG 46228723 IC50 = 11900 nM T99799 CK62AH 46228724 IC50 = 11900 nM T99799 C20GZR 46228760 IC50 = 3520 nM T99799 C4O9CE 46228761 IC50 = 99800 nM T99799 CLUW07 46228762 IC50 = 10000 nM T99799 CJ5YZ9 46228787 IC50 = 2700 nM T99799 CJ2D5H 46228788 IC50 = 7700 nM T99799 CJG67U 46228789 IC50 = 20500 nM T99799 CTBX50 46228809 IC50 = 33000 nM T99799 C6O3FS 46228810 IC50 = 90300 nM T99799 C0PHL3 46228811 IC50 = 135000 nM T99799 C9IE5S 46228812 IC50 = 72800 nM T99799 C7POL5 46228839 IC50 = 8050 nM T99799 C1E3LQ 46228840 IC50 = 5010 nM T99799 CEBO01 46229144 Ki = 9 nM T99799 CEL2V1 46229162 Ki = 250 nM T99799 C7Q6RX 46231880 IC50 = 5000 nM T99799 CH4K6D 46232763 IC50 = 10250 nM T99799 CH9EG0 46232810 IC50 = 4800 nM T99799 CI3DT1 46232813 IC50 = 52 nM T99799 C6C1ER 46232814 IC50 = 201 nM T99799 C0VIS5 46854881 IC50 = 20 nM T99799 CD0Q4G 46855034 IC50 = 6.5 nM T99799 CBO8D7 46863225 IC50 = 7900 nM T99799 CJ16FO 46866088 IC50 = 800 nM T99799 CG0UA1 46877971 IC50 = 1300 nM T99799 CX7J9D 46880263 IC50 = 2360000 nM T99799 CM6PJ3 46880264 IC50 = 1270000 nM T99799 C61VGD 46880266 IC50 = 1380000 nM T99799 C5G4FV 46880955 IC50 = 78000 nM T99799 CHNP43 46888221 IC50 > 200000 nM T99799 CZQL62 46897981 IC50 = 210 nM T99799 C4TWY7 46897983 IC50 = 140 nM T99799 CDG49K 46897985 IC50 = 43 nM T99799 CA7CK3 46897987 IC50 = 51 nM T99799 CY7ZW5 46937311 IC50 = 0.86 nM T99799 CXJ04C 49796971 IC50 = 406 nM T99799 CC86IT 49799305 IC50 = 130 nM T99799 CZYU91 49801688 IC50 = 4480 nM T99799 C35VYE 49845186 IC50 = 2450000 nM T99799 C4FHO0 49845187 IC50 = 1620000 nM T99799 CA9E5S 49845368 IC50 = 2140000 nM T99799 C6SE1Z 49845372 IC50 = 430000 nM T99799 C6BC2U 49845373 IC50 = 1580000 nM T99799 C7IJ3C 49857726 Ki > 100000 nM T99799 C04NYX 49857906 Ki > 100000 nM T99799 CDT4Y6 49857907 Ki > 100000 nM T99799 C5XS3G 49857908 Ki > 100000 nM T99799 CHRB62 49857909 Ki > 100000 nM T99799 CV7J6X 49857910 Ki > 100000 nM T99799 CYU39N 49857911 Ki > 100000 nM T99799 C5WZL0 49857912 Ki > 100000 nM T99799 CCG80U 49858100 Ki > 100000 nM T99799 CCN05H 49858101 Ki > 100000 nM T99799 C2OK0N 50874404 IC50 > 50000 nM T99799 CJE91N 50874405 IC50 > 50000 nM T99799 CTQX80 50942800 IC50 = 60 nM T99799 C8DS0J 50942802 IC50 = 16 nM T99799 CA43KF 51026481 IC50 = 170 nM T99799 C9VXK3 51039357 IC50 = 64000 nM T99799 CU36CR 51039359 IC50 = 25000 nM T99799 C8X5WJ 51039361 IC50 = 600 nM T99799 C1BA7H 51039363 IC50 = 1000 nM T99799 C4RQZ0 51039365 IC50 = 4000 nM T99799 C61UMV 51042596 IC50 = 154000 nM T99799 C2I3RA 51346780 IC50 = 1600 nM T99799 C4MH6G 51346832 IC50 = 400 nM T99799 C9AZ3J 51357040 IC50 > 10000 nM T99799 C8T1BE 51357043 IC50 > 10000 nM T99799 C3BRM2 51357044 IC50 > 10000 nM T99799 CIZ96K 51357316 IC50 > 10000 nM T99799 C5RXF2 51357319 IC50 > 10000 nM T99799 C6G9SM 51357595 Ki = 2100 nM T99799 C1R0DP 51357597 Ki = 79 nM T99799 CU0I5S 51357598 Ki = 2600 nM T99799 CE3H6X 51357599 Ki = 380 nM T99799 CGV79B 51357600 IC50 > 10000 nM T99799 C6S1KB 51357868 IC50 > 10000 nM T99799 C7QPU6 52110752 IC50 = 22000 nM T99799 CD52WQ 52111959 IC50 = 11400 nM T99799 C0LG4K 52899556 IC50 = 58600 nM T99799 CEGS83 52940502 IC50 = 940 nM T99799 C5PJL4 52940842 IC50 = 97000 nM T99799 C3F7VC 52946604 IC50 = 230 nM T99799 CQRK41 52948055 IC50 = 64000 nM T99799 C3ORW4 52949034 IC50 = 920 nM T99799 C8ZKR5 52952236 IC50 = 36 nM T99799 C4JG6W 52952244 IC50 = 620 nM T99799 CIO3V4 52952919 IC50 = 35000 nM T99799 C61YEU 52952920 IC50 = 11000 nM T99799 C9T8YE 52952921 IC50 = 9700 nM T99799 CDYC75 52952922 IC50 = 21900 nM T99799 C4Z6WM 52952958 IC50 = 39000 nM T99799 C8XV3H 52993127 IC50 = 9010 nM T99799 CPMW48 53231243 IC50 = 209000 nM T99799 CD4NP3 53231341 IC50 = 144000 nM T99799 C6RE1G 53231342 IC50 = 145000 nM T99799 CK64RX 53231343 IC50 = 179000 nM T99799 C4VE2O 53231344 IC50 = 68000 nM T99799 CNC2D0 53231345 IC50 = 21000 nM T99799 C0Z3AM 53231442 IC50 = 34000 nM T99799 C5A3YX 53231443 IC50 = 10400 nM T99799 CPM56F 53231444 IC50 = 23000 nM T99799 CO40KS 53231445 IC50 = 24200 nM T99799 C5M0OA 53242257 Ki = 1740 nM T99799 C9EL0U 53306553 IC50 = 3326 nM T99799 C3DS7L 53316786 IC50 = 241000 nM T99799 C67YGU 53320725 IC50 = 150 nM T99799 CY9HE5 53320727 IC50 = 110 nM T99799 CF0AC4 53320729 IC50 = 19000 nM T99799 CY7J8V 53320731 IC50 = 1300 nM T99799 CXB5G7 53321044 IC50 > 10000 nM T99799 C0DUN8 53321516 IC50 = 3000 nM T99799 CFKJ51 53322024 Ki = 100 nM T99799 CH1O9A 53322846 IC50 = 700 nM T99799 C26USF 53323382 IC50 = 700 nM T99799 CZT5X1 53323384 IC50 = 2400 nM T99799 C2RJQ1 53324171 IC50 = 2600000 nM T99799 CE0W5F 53324336 IC50 = 1900 nM T99799 CM1KA7 53324700 IC50 = 5100 nM T99799 C1XL0O 53324702 IC50 = 4400 nM T99799 C4YWN2 53326005 IC50 = 600 nM T99799 CW8ZV1 53326729 IC50 = 2000 nM T99799 CK45JD 53361165 IC50 = 0.0449 nM T99799 CTSC36 53361167 IC50 = 0.0354 nM T99799 CIP6E3 53361169 IC50 = 0.0212 nM T99799 CWK2J9 54097201 IC50 = 8130 nM T99799 CDCR53 54577393 IC50 = 24.8 nM T99799 CUSF85 54577394 IC50 = 63.7 nM T99799 CVJA50 54577395 IC50 = 1660 nM T99799 CXOH83 54577607 IC50 = 28.6 nM T99799 CD8PN5 54580372 IC50 = 871000 nM T99799 CT2L8P 54580374 IC50 = 308000 nM T99799 C7DH8A 54580376 IC50 = 200 nM T99799 C1IE9P 54580388 IC50 = 501 nM T99799 C3ENI1 54580389 IC50 > 10000 nM T99799 CN20LZ 54581356 IC50 > 10000 nM T99799 C6KVB5 54581375 IC50 = 700 nM T99799 CBH4L1 54581388 IC50 > 1000 nM T99799 C23NPW 54582394 IC50 = 13000 nM T99799 CH60OU 54582403 IC50 > 10000 nM T99799 C1MZ0J 54582404 IC50 > 10000 nM T99799 CX8N5Y 54582406 IC50 > 10000 nM T99799 CXVQ08 54583385 IC50 = 1430 nM T99799 C7WS9L 54583386 IC50 = 333 nM T99799 C8NXY5 54583387 IC50 = 679 nM T99799 C21PHC 54584309 IC50 = 224 nM T99799 CZ8E5U 54584310 IC50 = 217 nM T99799 CH7JX8 54584326 IC50 = 20000 nM T99799 CZW86O 54584337 IC50 > 10000 nM T99799 CVB76W 54584338 IC50 = 554 nM T99799 CW8EU4 54585277 IC50 > 10000 nM T99799 C9VCF6 54585278 IC50 > 10000 nM T99799 C9ZSE5 54585303 IC50 = 32000 nM T99799 C2SQ7Y 54586227 IC50 = 5375 nM T99799 CNEB14 54586228 IC50 = 1343 nM T99799 C97ESH 54586244 IC50 = 400 nM T99799 CUR47F 54587253 IC50 = 477 nM T99799 CY9X6B 54587254 IC50 = 653 nM T99799 C0WMB8 54587272 IC50 = 48000 nM T99799 C8PH1A 54587274 IC50 = 800 nM T99799 CV3F8K 54587276 IC50 = 6000 nM T99799 C75HCV 54587283 IC50 > 10000 nM T99799 C9KL7N 54587284 IC50 = 2948 nM T99799 C3Y1NF 54604881 IC50 > 5000 nM T99799 C4JOA7 54753261 IC50 = 1100 nM T99799 CE1ZN5 54754513 IC50 > 200000 nM T99799 CQ1MY9 54768917 IC50 = 101 nM T99799 C61LVE 54768918 IC50 = 90.5 nM T99799 C6FD9U 54768919 IC50 = 42.8 nM T99799 CD19BL 54768920 IC50 = 38.1 nM T99799 CVQ80D 54768921 IC50 = 14.7 nM T99799 CSUP59 54768922 IC50 = 101 nM T99799 CAP3I8 54769156 IC50 = 7280 nM T99799 C9O1JY 54769157 IC50 = 41.4 nM T99799 CFYX02 56649564 IC50 = 8570 nM T99799 C9TNA0 56926078 IC50 = 3160 nM T99799 CH46AD 56926079 IC50 = 3580 nM T99799 CJ31RE 56930476 IC50 = 30.6 nM T99799 CNYF34 56930477 IC50 = 205000 nM T99799 C0J2NP 56930478 IC50 = 398 nM T99799 CDQ32W 56933910 IC50 = 3780 nM T99799 CXNJ86 56933912 IC50 = 119000 nM T99799 CLB67G 56934051 IC50 = 26100 nM T99799 C4ZBA5 56934056 IC50 > 100000 nM T99799 CMA7L0 56954888 IC50 = 0.08 nM T99799 C4M1ET 56954890 IC50 = 0.038 nM T99799 C8XCI0 56954891 IC50 = 0.1 nM T99799 CHV8U3 56954986 IC50 = 0.1 nM T99799 CV3X9D 56954987 IC50 = 0.1 nM T99799 C0JCZ2 56954989 IC50 = 15 nM T99799 CTB71C 56954996 IC50 = 0.15 nM T99799 C4A6LW 56955097 IC50 = 50 nM T99799 CC7Y5O 56955099 IC50 = 1.5 nM T99799 C25KBX 56955100 IC50 = 1.5 nM T99799 C9XO0M 56955109 IC50 = 1 nM T99799 COE65B 56955111 IC50 = 0.8 nM T99799 C4U9FZ 56955198 IC50 = 5 nM T99799 C9I3AY 56955199 IC50 = 2.5 nM T99799 C2EY4O 56955292 IC50 = 30 nM T99799 C2M6DQ 56955293 IC50 = 95 nM T99799 CHA1I9 57342686 IC50 > 3000000 nM T99799 CZBE16 57342689 IC50 = 375.9 nM T99799 CC76WY 57342690 IC50 = 42.6 nM T99799 CVK98Q 57383995 IC50 = 1.57 nM T99799 CHB7N4 57390352 IC50 > 200000 nM T99799 CNM3O8 57390398 IC50 = 656000 nM T99799 CZDN40 57391125 IC50 = 78800 nM T99799 COAM20 57392136 IC50 > 200000 nM T99799 C5D7HF 57396286 IC50 = 12.1 nM T99799 CJE63A 57397445 IC50 > 200000 nM T99799 CZ3KT7 57402629 IC50 > 200000 nM T99799 CPUM70 59740711 IC50 = 2030 nM T99799 CV2G0U 60144120 IC50 = 82000 nM T99799 CVO2Z4 60148583 IC50 = 549.2 nM T99799 C4F1PE 60165327 IC50 = 6.4 nM T99799 CO58SL 60661850 IC50 > 100000 nM T99799 C4KS0V 62707049 IC50 = 11.2 nM T99799 CNW04I 62707050 IC50 = 1.71 nM T99799 C1U2FD 62707051 IC50 = 27.6 nM T99799 CZV81L 64338500 IC50 > 100000 nM T99799 CYRU28 66573467 IC50 > 10000 nM T99799 CDVT38 66573526 IC50 > 10000 nM T99799 CSA1R0 66573527 IC50 > 10000 nM T99799 CN0H5V 66573528 IC50 = 9370 nM T99799 CE52KG 66573529 IC50 > 10000 nM T99799 CMXZ21 66573530 IC50 > 10000 nM T99799 CC9Z1H 66573531 IC50 > 10000 nM T99799 C3W0YV 66573584 IC50 > 10000 nM T99799 C9QK4S 66573585 IC50 > 10000 nM T99799 C32IQA 66573586 IC50 > 10000 nM T99799 C0YE1R 68259803 IC50 = 81600 nM T99799 CJ7M5L 70683121 IC50 = 74.2 nM T99799 C09ICA 70684451 IC50 = 211 nM T99799 CD16OS 70684889 IC50 = 1500 nM T99799 CPO69B 70685195 IC50 = 44.2 nM T99799 C9HE4I 70685196 IC50 = 51.3 nM T99799 CXY5N6 70686590 IC50 = 41.2 nM T99799 CN8XT5 70687043 IC50 = 260 nM T99799 C5WOI8 70689140 IC50 = 6600 nM T99799 C7LMF4 70689416 IC50 = 24.6 nM T99799 CE4OI8 70689417 IC50 = 75.2 nM T99799 CV1DC5 70689418 IC50 = 35.1 nM T99799 CU2XC0 70690775 IC50 = 137 nM T99799 C8RPA4 70692911 IC50 = 63.7 nM T99799 CC3Y2P 70692912 IC50 = 33.7 nM T99799 CW8AX2 70692913 IC50 = 1520 nM T99799 C6AHB9 70693333 IC50 > 10000 nM T99799 CA7CP6 70693341 IC50 = 580 nM T99799 C2LV8M 70694951 IC50 = 126 nM T99799 CC39LU 70695442 IC50 = 670 nM T99799 C1U2SF 70695443 IC50 = 1700 nM T99799 CF9EO8 70697005 IC50 = 77.8 nM T99799 CWO7H5 70697453 IC50 > 10000 nM T99799 CN93VA 71330901 IC50 = 4700 nM T99799 C7AJN9 71449137 IC50 = 16.4 nM T99799 CX8KG3 71449167 IC50 > 50000 nM T99799 CRC86Q 71449660 Ki = 56 nM T99799 CVF86W 71449711 IC50 = 400 nM T99799 C06WZI 71449712 IC50 = 1970 nM T99799 C24OJQ 71451471 Ki = 97 nM T99799 CVKC68 71451473 Ki = 93 nM T99799 C7NS9H 71451521 IC50 = 3180 nM T99799 CDES68 71451522 IC50 = 23000 nM T99799 CJ1AS9 71452935 IC50 = 61.2 nM T99799 C5CK7V 71453297 Ki = 55 nM T99799 CJD10W 71453346 IC50 = 136000 nM T99799 CYVB31 71453347 IC50 = 6600 nM T99799 CTJ6W4 71453348 IC50 = 880 nM T99799 CN14WJ 71453349 IC50 = 43900 nM T99799 CJ4B5X 71453350 IC50 = 2510 nM T99799 CHGF12 71453367 IC50 = 1890 nM T99799 C28XSH 71454519 IC50 = 31.1 nM T99799 C2JYF6 71455057 IC50 = 88900 nM T99799 C4JDI7 71455058 IC50 = 2880 nM T99799 CL4F6Z 71455059 IC50 = 48 nM T99799 CAJ7O6 71456744 IC50 = 20360 nM T99799 CL02JI 71456801 Ki = 166 nM T99799 CC7F6N 71456803 Ki = 82 nM T99799 C2B8LY 71456805 Ki = 99 nM T99799 CA93KH 71456856 IC50 = 7470 nM T99799 C1D6KG 71456857 IC50 = 60100 nM T99799 CP1OY9 71456858 IC50 = 89100 nM T99799 CP4K8E 71456859 IC50 = 21000 nM T99799 C10XZB 71458090 IC50 > 50000 nM T99799 C3ZU1K 71458289 IC50 = 50.1 nM T99799 CV5TX6 71458713 IC50 = 55600 nM T99799 CH7L4U 71458714 IC50 = 81200 nM T99799 C35XHD 71458715 IC50 = 1810 nM T99799 C3ASY5 71458716 IC50 = 3010 nM T99799 C0YS7T 71460136 IC50 = 9.2 nM T99799 CXHM16 71460484 Ki = 2360 nM T99799 C2JBI7 71462190 Ki = 66 nM T99799 CTY0B6 71462239 IC50 = 3000 nM T99799 CBM3S6 71462240 IC50 = 9420 nM T99799 C5YHW6 71462241 IC50 = 1370 nM T99799 C7DQL5 71475219 IC50 = 499000 nM T99799 C8ZDA2 71492183 IC50 = 375300 nM T99799 CLN29O 71587645 Ki = 0.131 nM T99799 CD5K9Y 71602709 IC50 = 8270 nM T99799 CLGH80 71653617 IC50 = 108.97 nM T99799 CEI5B1 71653619 IC50 = 57.3 nM T99799 CC45NP 71653620 IC50 = 82.34 nM T99799 CA81JD 71653759 IC50 = 30.47 nM T99799 CW9EZ1 71653760 IC50 = 120.13 nM T99799 CIFJ03 71653761 IC50 = 92.42 nM T99799 C1LVE7 71653762 IC50 = 37.57 nM T99799 CRYS21 71653918 IC50 = 67.31 nM T99799 C25PJH 71653919 IC50 = 61.69 nM T99799 CJ9LX8 71653920 IC50 = 7.1 nM T99799 CY9Z1K 71654077 IC50 = 76.89 nM T99799 CMFG63 71654078 IC50 = 58 nM T99799 CSW15Q 71654079 IC50 = 29.28 nM T99799 COH09E 71654080 IC50 = 34.75 nM T99799 C7Q5ON 71654239 IC50 = 55.25 nM T99799 CSF8E7 71654240 IC50 = 35.98 nM T99799 CS5M3R 71654241 IC50 = 29.56 nM T99799 CT8WV6 71654242 IC50 = 12.44 nM T99799 CFMB35 71723450 IC50 > 100000 nM T99799 CV16HS 71723451 IC50 > 100000 nM T99799 C7U5ER 71723452 IC50 = 71920 nM T99799 CF2VL4 71723589 IC50 = 2260 nM T99799 COT21H 71723590 IC50 > 100000 nM T99799 C9RLM5 71769057 Ki = 16820 nM T99799 C9NYJ2 71770939 Ki = 624425 nM T99799 CN06CX 71770940 Ki = 282620 nM T99799 C4R9EZ 72374595 IC50 = 8130 nM T99799 CK38PO 72374596 IC50 > 10000 nM T99799 C0FN4W 72374597 IC50 > 10000 nM T99799 C9LNA8 72376170 IC50 = 9410 nM T99799 CULW84 72376171 IC50 = 5620 nM T99799 CY19TH 72376172 IC50 = 8390 nM T99799 C45BXP 72543919 IC50 = 22500 nM T99799 C78ZPH 72544154 IC50 = 14700 nM T99799 CKAG40 72544155 IC50 = 360 nM T99799 CPH96F 72544156 IC50 = 18700 nM T99799 CE49KY 72544381 IC50 > 20000 nM T99799 CTW28Y 72544382 IC50 = 16400 nM T99799 C6TQ7M 72545286 IC50 = 9980 nM T99799 CBL6J5 72545287 IC50 = 7770 nM T99799 CKY67A 72724835 IC50 = 1000 nM T99799 C59UPS 72724837 IC50 = 7700 nM T99799 CA16UV 72724839 IC50 = 350 nM T99799 CTB2A1 72724841 IC50 = 370 nM T99799 C02IHQ 72724843 IC50 = 700 nM T99799 CGJ2T1 72724905 IC50 = 2200 nM T99799 C5Z4BW 72724907 IC50 = 2000 nM T99799 CJA54D 72724909 IC50 = 1700 nM T99799 C3OUZ2 72724911 IC50 = 3200 nM T99799 CY2M3K 72724913 IC50 = 900 nM T99799 CPWA14 72724915 IC50 = 680 nM T99799 C1LH5Z 72725438 Ki = 0.06 nM T99799 C6CJT1 72725439 Ki = 8.26 nM T99799 C3K0SD 72725440 Ki = 40.9 nM T99799 CS1TQ7 72725488 Ki = 61.77 nM T99799 C9ZB1M 72725489 Ki = 21.26 nM T99799 C53XHE 73346133 IC50 = 470 nM T99799 C9RWV8 73352248 IC50 > 10000 nM T99799 COKX05 73352249 IC50 > 10000 nM T99799 C45GXL 73356781 IC50 > 10000 nM T99799 CGD8R4 73671789 IC50 = 2100 nM T99799 CV13PU 76310709 IC50 > 10000 nM T99799 CZ49PQ 76311731 IC50 = 26000 nM T99799 CGI2O5 76317912 IC50 > 25000 nM T99799 C1I2UO 76317913 IC50 = 970 nM T99799 CE5M1O 76317914 IC50 > 10000 nM T99799 CC1PL3 76318071 IC50 = 1370 nM T99799 C4M8ZY 76321622 IC50 > 10000 nM T99799 CSXH87 76321623 Ki = 220 nM T99799 C1W8HB 76325234 Ki = 1200 nM T99799 CO05NW 76325235 Ki = 1000 nM T99799 C5AV9G 76328789 Ki = 28 nM T99799 C4QH5I 76328790 IC50 > 10000 nM T99799 C30AMV 76328791 IC50 > 100000 nM T99799 CB1KJ6 76328792 Ki = 2900 nM T99799 CEKP26 76328944 IC50 = 2590 nM T99799 CTG51J 76336093 IC50 > 10000 nM T99799 C48RZI 76336227 IC50 = 920 nM T99799 C57UTS 77108165 IC50 = 3700 nM T99799 C0JCK7 77461631 IC50 = 7224 nM T99799 C7GX5I 78350462 IC50 = 540 nM T99799 CA3YL2 78426937 IC50 > 40000 nM T99799 CR0H5Q 78427074 IC50 > 40000 nM T99799 C2ZOJ4 78427075 IC50 = 32000 nM T99799 CJCL87 78427076 IC50 = 15900 nM T99799 CH3NJ9 78427077 IC50 > 40000 nM T99799 CR84AG 78427078 IC50 > 40000 nM T99799 CV9DO7 78427079 IC50 > 40000 nM T99799 C4US9B 78427204 IC50 = 3100 nM T99799 CS0N1V 78427205 IC50 = 18900 nM T99799 CG46NS 78427206 IC50 > 40000 nM T99799 C3WL0E 78427207 IC50 = 14600 nM T99799 CK5X0H 78427208 IC50 = 12100 nM T99799 CN6L8C 78427209 IC50 = 21300 nM T99799 CCE8Q9 78427338 IC50 = 6500 nM T99799 C0CL4Y 80772460 IC50 = 5000 nM T99799 CI5GO1 83453608 IC50 = 18000 nM T99799 C5MC7H 85470203 IC50 = 5990 nM T99799 CHXN26 85852196 Ki = 341000 nM T99799 CB3ZI5 86294786 IC50 = 5830 nM T99799 CXC80P 86581945 IC50 = 9200 nM T99799 C8CF5A 88749792 IC50 > 100000 nM T99799 CRZ0W3 90356636 IC50 = 14900 nM T99799 CI3ZW5 90356648 IC50 > 40000 nM T99799 C85UDM 90356741 IC50 > 40000 nM T99799 C2Z5FB 90356750 IC50 > 40000 nM T99799 CYB89Q 90356760 IC50 = 14100 nM T99799 CW8N4S 90356765 IC50 > 40000 nM T99799 C3NKB2 90356879 IC50 = 29200 nM T99799 CO1RJ4 90356882 IC50 = 27800 nM T99799 C9UI0O 90356903 IC50 > 40000 nM T99799 CO2HX6 90356923 IC50 = 17600 nM T99799 C52SQL 90356955 IC50 > 40000 nM T99799 C5YD7M 90356964 IC50 = 33200 nM T99799 C31XOK 90357088 IC50 > 40000 nM T99799 C0P3IL 90357101 IC50 > 40000 nM T99799 CR54TH 90357102 IC50 = 17900 nM T99799 CBJ4I2 90357105 IC50 > 40000 nM T99799 CDXO02 90357107 IC50 = 24700 nM T99799 CY9T0A 90357109 IC50 > 40000 nM T99799 CWKM49 90357121 IC50 = 21100 nM T99799 CZ7CG4 90357147 IC50 = 23400 nM T99799 C1FKL7 90357154 IC50 > 40000 nM T99799 C1LO9P 90357159 IC50 = 20100 nM T99799 CYDQ90 90357180 IC50 > 40000 nM T99799 C3I9SK 90357196 IC50 = 18400 nM T99799 CSY64P 90357367 IC50 = 4200 nM T99799 C3YJ1K 90643449 IC50 = 333300 nM T99799 CJTA92 90643450 IC50 = 362300 nM T99799 CP72GI 90643451 IC50 = 384600 nM T99799 C5SAX0 90643452 IC50 = 409000 nM T99799 CZTO98 90643453 IC50 = 430000 nM T99799 CL4Z8B 90643454 IC50 = 451000 nM T99799 C0LKB7 90643455 IC50 = 452000 nM T99799 C6RY4Q 90643456 IC50 = 454500 nM T99799 CW28SA 90643457 IC50 = 500000 nM T99799 CO3G4W 90643458 IC50 = 512000 nM T99799 CWG1P9 90643459 IC50 = 568000 nM T99799 CS0N9O 90643460 IC50 = 585000 nM T99799 CN8XQ5 90643461 IC50 = 100 nM T99799 CR67MP 90643462 IC50 = 248000 nM T99799 C0DIJ2 90643463 IC50 = 294000 nM T99799 C1E8XY 90643464 IC50 = 295000 nM T99799 CJW74Q 90643465 IC50 = 297600 nM T99799 C6Z3CW 90643468 IC50 = 19700 nM T99799 CHW4X8 90643469 IC50 = 42400 nM T99799 CU8A1S 90643470 IC50 = 43600 nM T99799 CEAB94 90643471 IC50 = 65500 nM T99799 CUO8H3 90643472 IC50 = 83300 nM T99799 CTVJ69 90645106 IC50 = 43660 nM T99799 CYW8G5 90645107 IC50 = 38530 nM T99799 C1R6LU 90645108 IC50 = 12340 nM T99799 C5U8JA 90645109 IC50 > 100000 nM T99799 C8CKM6 90645110 IC50 = 65270 nM T99799 CYN86M 90645111 IC50 = 88930 nM T99799 C3EAW0 90645112 IC50 = 14660 nM T99799 C4XF1V 90645113 IC50 > 100000 nM T99799 C30WLJ 90645114 IC50 > 100000 nM T99799 CG6YO8 90645115 IC50 > 100000 nM T99799 CJZ4X5 90645116 IC50 > 100000 nM T99799 CO20MQ 90645117 IC50 = 19740 nM T99799 C8QHF2 90645118 IC50 = 22650 nM T99799 CVPN52 90645119 IC50 > 100000 nM T99799 CXHK56 90645120 IC50 > 100000 nM T99799 CF4EB2 90645121 IC50 > 100000 nM T99799 CB2E7N 90645122 IC50 > 100000 nM T99799 CR2VS4 90645123 IC50 > 100000 nM T99799 C1ZYO3 90645124 IC50 > 100000 nM T99799 C2CI1S 90645125 IC50 > 100000 nM T99799 C40YGU 90645126 IC50 > 100000 nM T99799 C4R7BX 90645127 IC50 > 100000 nM T99799 CMN7Z9 90645128 IC50 > 100000 nM T99799 C62RBA 90645129 IC50 = 66750 nM T99799 CXU48E 90645130 IC50 = 56920 nM T99799 CYG4D2 90645131 IC50 > 100000 nM T99799 CPM6V1 90645132 IC50 > 100000 nM T99799 CP1OU8 90645133 IC50 > 100000 nM T99799 CAB7V8 90654202 IC50 = 4.28 nM T99799 CX03IG 90654705 IC50 = 3850 nM T99799 C93PIK 90654706 IC50 = 1250 nM T99799 CWLF50 90654707 IC50 = 5190 nM T99799 CP5T0F 90654708 IC50 = 7650 nM T99799 CP4U3I 90654791 IC50 = 36200 nM T99799 C62CPS 90654792 IC50 = 32100 nM T99799 CLI41J 90654793 IC50 = 39150 nM T99799 CNJ69Y 90654795 IC50 = 52760 nM T99799 CWQ16H 90654796 IC50 = 39410 nM T99799 CD1FR7 90654797 IC50 = 18010 nM T99799 CWF6X2 90654981 IC50 = 5.66 nM T99799 CMC46P 90655184 IC50 = 950 nM T99799 C12GDL 90655186 IC50 = 1070 nM T99799 C36VCM 90655188 IC50 = 1460 nM T99799 CL7PI9 90655190 IC50 = 350 nM T99799 CZ18NX 90655191 IC50 = 620 nM T99799 CH7C4F 90655192 IC50 = 265 nM T99799 CMJ31X 90655193 IC50 = 513 nM T99799 C3IZ2O 90655195 IC50 = 1100 nM T99799 CG69TU 90655196 IC50 = 645 nM T99799 C6WH0F 90655198 IC50 = 510 nM T99799 CT2N6S 90656307 IC50 = 23730 nM T99799 CTXS90 90656308 IC50 = 10590 nM T99799 CHJ71K 90656309 IC50 = 15900 nM T99799 C1FSU2 90656310 IC50 = 12900 nM T99799 CMAJ10 90656311 IC50 = 21710 nM T99799 CY0KN8 90656312 IC50 = 9290 nM T99799 CF9A7K 90656313 IC50 = 16700 nM T99799 C2I0ZP 90656314 IC50 = 3430 nM T99799 CKXS95 90656315 IC50 = 11170 nM T99799 CP4D2I 90656316 IC50 = 6020 nM T99799 CDV62L 90656317 IC50 = 6420 nM T99799 C2E0NT 90656318 IC50 = 3250 nM T99799 CS4ZQ0 90656319 IC50 = 2270 nM T99799 CNCZ35 90663111 IC50 > 50000 nM T99799 CP48CG 90663114 IC50 > 50000 nM T99799 C6JS8W 90664279 IC50 = 700 nM T99799 CY86BC 90664299 IC50 = 1931 nM T99799 C7NGZ1 90664300 IC50 = 218 nM T99799 C1KOL2 90664301 IC50 = 1076 nM T99799 C30SQY 90664402 IC50 = 331 nM T99799 CKU86A 90664403 IC50 = 1391 nM T99799 CM4NF3 90664404 IC50 = 1622 nM T99799 CKL69C 90664470 IC50 = 87.1 nM T99799 CL65ZG 90664552 IC50 = 586 nM T99799 C0GN8Y 90664609 IC50 = 43.3 nM T99799 C05QSY 90664655 Ki = 379700 nM T99799 CPE7N6 90664658 IC50 = 88.7 nM T99799 CYGT83 90664665 IC50 = 234 nM T99799 CO82LG 90664779 IC50 = 136 nM T99799 C90OVC 90664784 IC50 = 1074 nM T99799 C4EA8P 90664797 IC50 = 55 nM T99799 C7H6ZG 90664851 IC50 = 26.6 nM T99799 C3AON4 90664852 IC50 = 73.3 nM T99799 CI0NQ2 90664853 IC50 = 86.8 nM T99799 CLQ1F4 90664854 IC50 = 47.4 nM T99799 CFK51Z 90664907 IC50 = 66.3 nM T99799 CI1T4S 90664976 IC50 = 133 nM T99799 CXB25V 90664977 IC50 = 27.2 nM T99799 C1DN7L 90664978 IC50 = 76.6 nM T99799 CFPS72 90665034 Ki = 273400 nM T99799 CW36ZP 90665154 IC50 = 72.7 nM T99799 C80QZK 90665217 IC50 = 139 nM T99799 CB70OR 90667344 IC50 = 30000 nM T99799 C17ZXD 90667346 IC50 = 6700 nM T99799 C2JT9Z 90667348 IC50 = 65000 nM T99799 C8SUR1 90667350 IC50 = 10000 nM T99799 CTDR94 90667352 IC50 = 60000 nM T99799 CYIJ47 90667354 IC50 > 1000000 nM T99799 C6J7ZA 90667356 IC50 = 4200 nM T99799 CTWS98 90667358 IC50 = 1600 nM T99799 C1PY0T 90676323 IC50 = 11700 nM T99799 CQ76YM 90679728 IC50 = 34673.69 nM T99799 C9AM2Q 90679729 IC50 = 21877.62 nM T99799 CUDM30 90679730 IC50 = 9772.37 nM T99799 C9PX6B 90679731 IC50 = 1047.13 nM T99799 C1S8AL 91031465 IC50 = 220 nM T99799 CG9JP4 91689645 IC50 = 3600 nM T99799 C7C9RB 91689712 IC50 = 30800 nM T99799 C8NC7S 91689713 IC50 = 32600 nM T99799 CAM0G8 91864546 IC50 = 2.18 nM T99799 CUPK70 91885433 IC50 = 3900 nM T99799 C5RF6O 101077957 IC50 > 30000 nM T99799 C4HLR3 101528287 IC50 > 30000 nM T99799 C20CYQ 101879984 IC50 = 585 nM T99799 C5V2JH 101886788 IC50 = 256 nM T99799 CLO03N 101886789 IC50 = 41.4 nM T99799 CF6EI0 101886790 IC50 = 5.45 nM T99799 C52VTG 101886792 IC50 = 19.1 nM T99799 CV3A0F 101886793 IC50 = 501 nM T99799 CI2U0Y 101886794 IC50 = 197 nM T99799 C56IGC 101886796 IC50 = 258 nM T99799 C6W2JF 101898808 Ki = 16.1 nM T99799 C81WRJ 101910778 IC50 = 4900 nM T99799 CDBZ20 102189779 IC50 = 2844 nM T99799 C1PAK7 102257397 IC50 = 13460 nM T99799 C71RIU 102257398 IC50 = 8930 nM T99799 C4XMG6 102257401 IC50 = 10420 nM T99799 C0NV1I 102286159 IC50 > 10000 nM T99799 C4LJ9O 102369422 IC50 = 267 nM T99799 CY93VO 102369423 IC50 = 328 nM T99799 CYG4M5 102484612 IC50 > 50000 nM T99799 CDRX58 118622604 IC50 > 40000 nM T99799 CP5Z8M 118622610 IC50 = 16200 nM T99799 C7TZ2R 118622611 IC50 = 12700 nM T99799 CRW07P 118622616 IC50 = 8500 nM T99799 CIP1L6 118706200 IC50 = 99 nM T99799 C9M3EL 118709900 IC50 = 765 nM T99799 CMWO04 118709901 IC50 = 228 nM T99799 C39HSZ 118709912 IC50 = 2030 nM T99799 CI38GE 118709913 IC50 = 2380 nM T99799 CH5V0G 118709914 IC50 = 2230 nM T99799 CBP3S5 118709915 IC50 = 12600 nM T99799 CT1J4G 118709916 IC50 = 827 nM T99799 C4IZB0 118709917 IC50 = 1420 nM T99799 C7JDT6 118709918 IC50 = 5620 nM T99799 CEY60K 118709968 IC50 = 286 nM T99799 C8GS0O 118709970 IC50 = 120 nM T99799 CAGS07 118709972 IC50 = 205 nM T99799 C40GLT 118709974 IC50 = 337 nM T99799 C1J0IZ 118711805 Ki = 31.7 nM T99799 C8D5HF 118711806 Ki = 29.8 nM T99799 CLG7K5 118711807 Ki = 34 nM T99799 CQB1O3 118711808 Ki = 32.4 nM T99799 C5C3XE 118711809 Ki = 8.1 nM T99799 C3H2YI 118711810 Ki = 32.5 nM T99799 COUQ50 118711811 Ki = 20.2 nM T99799 COSI80 118711812 Ki = 23.7 nM T99799 CJG10W 118711813 Ki = 23.2 nM T99799 CNH93M 118711814 Ki = 31.2 nM T99799 C2Q8IE 118711815 Ki = 17.5 nM T99799 C3C0QD 118711816 Ki = 20 nM T99799 CG62FL 118711817 Ki = 35 nM T99799 C9U5SV 118712170 Ki = 34.5 nM T99799 C9KUS7 118712171 Ki = 50.9 nM T99799 CJH4K5 118712172 Ki = 37.5 nM T99799 CB74FU 118712173 Ki = 40 nM T99799 C1J5NW 118715681 IC50 = 79900 nM T99799 C2YJB1 118715683 IC50 = 70700 nM T99799 CO98FC 118715684 IC50 = 3020 nM T99799 C0JPI2 118715685 IC50 = 25400 nM T99799 CAI03B 118715686 IC50 = 15900 nM T99799 CVN98D 118715709 IC50 = 32290 nM T99799 CG78ML 118715710 IC50 = 11750 nM T99799 CBO21H 118715711 IC50 = 17420 nM T99799 C5JO1E 118715712 IC50 = 20120 nM T99799 CK8MI7 118715713 IC50 = 10240 nM T99799 C5S7WZ 118715714 IC50 = 26330 nM T99799 CN6QV9 118715715 IC50 = 18470 nM T99799 CF0RX8 118715716 IC50 = 52580 nM T99799 C6MD2K 118715717 IC50 = 10130 nM T99799 C57BFX 118715718 IC50 = 8840 nM T99799 C1EJ5Q 118715719 IC50 = 39650 nM T99799 CQ92DR 118715720 IC50 = 40740 nM T99799 CRD9N0 118715721 IC50 = 279110 nM T99799 C6T0HL 118715722 IC50 = 68250 nM T99799 CQS06R 118715723 IC50 = 41910 nM T99799 C31XUV 118715724 IC50 = 96920 nM T99799 C3ZO6M 118715725 IC50 = 75090 nM T99799 CV98EO 118718831 IC50 = 1800 nM T99799 CLE2S7 118720934 IC50 = 982 nM T99799 C23AHU 118720935 IC50 = 742 nM T99799 CJWC73 118720936 IC50 = 181 nM T99799 CCSQ94 118721626 IC50 = 635 nM T99799 CL7JH8 118721627 IC50 = 14.5 nM T99799 CK2G3V 118721628 IC50 = 1280 nM T99799 CU83LO 118721629 IC50 = 329 nM T99799 CJ3S7L 118721630 IC50 = 970 nM T99799 C4F0TD 118721871 IC50 = 742 nM T99799 C5MR9S 118721872 IC50 = 287 nM T99799 CK85GL 118721873 IC50 = 234 nM T99799 CRTA65 118721874 IC50 = 96.1 nM T99799 C6HM0O 118721875 IC50 = 47.8 nM T99799 C0C6VE 118724841 IC50 = 5080 nM T99799 CHX5E4 118724846 IC50 = 2000 nM T99799 C3MX8I 118724859 IC50 = 930 nM T99799 C5P3GX 118725584 IC50 = 3000 nM T99799 C4N1ZC 118725585 IC50 = 1200 nM T99799 C4SK9H 118725586 IC50 = 7000 nM T99799 CI58BM 118725587 IC50 = 15000 nM T99799 C92JNZ 118725588 IC50 = 61000 nM T99799 CAK26D 118725589 IC50 = 161000 nM T99799 C3OR9J 118725590 IC50 = 210000 nM T99799 C8ZG3S 118727884 IC50 = 550 ug.mL-1 T99799 CXOA52 118730192 IC50 = 5900 nM T99799 C27ZWI 118730193 IC50 = 7100 nM T99799 CEQ56Z 118730194 IC50 = 7300 nM T99799 C3D6VY 118730195 IC50 = 40600 nM T99799 CJ2P9D 118730196 IC50 = 9700 nM T99799 CI2X8N 118730197 IC50 = 31200 nM T99799 C07TJO 118732687 IC50 = 56.3 nM T99799 CFN57B 118732688 IC50 = 5.2 nM T99799 C1UWN7 118732689 IC50 = 10.2 nM T99799 C2LJX1 118732690 IC50 = 20.5 nM T99799 C1GS6P 118732691 IC50 = 19.2 nM T99799 CS73OE 118732692 IC50 = 34.7 nM T99799 C62UPS 118732693 IC50 = 110.1 nM T99799 CNB83Q 118734712 IC50 = 124.32 nM T99799 CX80VO 118734713 IC50 = 112.72 nM T99799 C87YTM 118736706 IC50 > 5000 nM T99799 C4CTX6 118736714 IC50 > 5000 nM T99799 CMB54K 118736716 IC50 > 5000 nM T99799 COS59D 118736718 IC50 > 5000 nM T99799 CIB78Z 118736720 IC50 = 2400 nM T99799 C2PO6M 118736722 IC50 = 3500 nM T99799 C0YHI7 122180159 IC50 > 30000 nM T99799 C5K0RY 122180160 Ki = 4780 nM T99799 C71TKE 122180161 IC50 > 30000 nM T99799 C9QKP3 122180162 IC50 = 420 nM T99799 CQL13W 122180163 IC50 = 1370 nM T99799 CMR72I 122180164 IC50 > 30000 nM T99799 C1X9KB 122180406 IC50 = 950 nM T99799 CMC26Y 122180416 IC50 = 950 nM T99799 CEJ8S0 122180431 IC50 = 890 nM T99799 CKM1E7 122180462 IC50 = 9300 nM T99799 CH36VG 122182060 IC50 = 2140 nM T99799 C4PB1D 122182066 IC50 = 215 nM T99799 CDI8W2 122186374 IC50 = 128740 nM T99799 CK0WP5 122186375 IC50 = 110530 nM T99799 CA7U0N 122186376 IC50 = 187540 nM T99799 CO8V2R 122186377 IC50 = 119210 nM T99799 CE67WU 122186379 IC50 = 118540 nM T99799 C6JYH5 122186381 IC50 = 296530 nM T99799 CLTA13 122186382 IC50 = 105230 nM T99799 C1FKJ5 122186383 IC50 = 106410 nM T99799 C8NRX7 122186486 IC50 = 99740 nM T99799 CMCJ76 122186487 IC50 = 89240 nM T99799 CS5C0T 122186488 IC50 = 151870 nM T99799 C9WA3O 122186489 IC50 = 81410 nM T99799 C8KFR9 122186490 IC50 = 26530 nM T99799 CV4EJ3 122186491 IC50 = 151350 nM T99799 CU08GD 122186492 IC50 = 4520 nM T99799 CI7UZ4 122186493 IC50 = 44830 nM T99799 CKYL61 122186494 IC50 = 5310 nM T99799 CGC6T5 122186495 IC50 = 140930 nM T99799 CDU7H8 122186496 IC50 = 78020 nM T99799 C0JK8P 122186497 IC50 = 491730 nM T99799 C1T7UF 122186498 IC50 = 25910 nM T99799 C21LZX 122186499 IC50 = 187540 nM T99799 CZ38FY 122186500 IC50 = 160950 nM T99799 C8CGX0 122186502 IC50 = 103430 nM T99799 CC28ZL 122186503 IC50 = 167820 nM T99799 CD37LR 122186505 IC50 = 75890 nM T99799 CP4V8H 122191089 IC50 = 1200 nM T99799 C7OGL4 122191091 IC50 = 10000 nM T99799 C73UCL 122191093 IC50 = 20000 nM T99799 C16CXB 122193107 IC50 = 280 nM T99799 C0Q6AY 122193108 IC50 = 340 nM T99799 CM8C5G 122193110 IC50 = 2800 nM T99799 CBQW34 122193112 IC50 = 4100 nM T99799 CAXZ47 122193114 IC50 = 5100 nM T99799 C0ASQ2 122193116 IC50 = 4800 nM T99799 CXN7T8 122193118 IC50 = 5800 nM T99799 CDKJ53 122193120 IC50 = 8900 nM T99799 C6S7CV 122193124 IC50 = 6800 nM T99799 CL8J3Z 122193126 IC50 = 7900 nM T99799 CZ96MQ 122193128 IC50 = 7500 nM T99799 CCZJ35 122193130 IC50 = 80 nM T99799 C7N1BE 122193132 IC50 = 2300 nM T99799 C0FJ1G 122193134 IC50 = 1100 nM T99799 CSU6Q5 122193237 IC50 = 710 nM T99799 CSY2D4 122193239 IC50 = 860 nM T99799 C5VTJ4 122193241 IC50 = 720 nM T99799 C5XAM3 122193243 IC50 = 650 nM T99799 CC7E1R 122194787 IC50 = 1300 nM T99799 CNH49U 122194788 IC50 = 620 nM T99799 CLG31E 122194789 IC50 = 290 nM T99799 CLOD26 122194790 IC50 = 400 nM T99799 CY3EJ9 122194791 IC50 = 690 nM T99799 CI7Q9F 122194792 IC50 = 700 nM T99799 C9C7VG 122194793 IC50 = 1530 nM T99799 C2A4ES 122194881 IC50 = 80 nM T99799 CI2K5Z 122194882 IC50 = 20 nM T99799 C1E3LP 122194883 IC50 = 770 nM T99799 C4A8JM 122194884 IC50 = 90 nM T99799 CR79OE 122194885 IC50 = 130 nM T99799 CZ8L9J 122194886 IC50 = 400 nM T99799 CK7B8R 122194887 IC50 = 700 nM T99799 CSNM01 122194888 IC50 = 54 nM T99799 C5JXL2 122199175 IC50 = 20 nM T99799 CEX9B4 122199179 IC50 = 1400 nM T99799 CPJ2K1 122199184 IC50 = 1900 nM T99799 C3N9DJ 122199186 IC50 = 70 nM T99799 C1T5SW 122199188 IC50 = 1600 nM T99799 CJV5B8 122387041 IC50 = 5000 nM T99799 CI89OZ 122387042 IC50 = 5000 nM T99799 CYWM69 122387043 IC50 = 11000 nM T99799 CFVL05 122387044 IC50 = 38000 nM T99799 CFI4B3 122387045 IC50 = 9600 nM T99799 CNS65E 122387046 IC50 = 11100 nM T99799 C6BG0C 122581932 Ki = 1.71 nM T99799 C50XJY 122581936 IC50 = 4.9 nM T99799 CQ8MG5 122581957 IC50 = 1.03 nM T99799 CO01UP 127025001 IC50 = 2670 nM T99799 CT6H9W 127025002 IC50 = 1680 nM T99799 C2Q8FW 127025129 IC50 = 2800 nM T99799 CAB51G 127025336 IC50 = 15280 nM T99799 CO3NW2 127025337 IC50 = 16250 nM T99799 CHW76D 127025338 IC50 = 12340 nM T99799 C06WQV 127025339 IC50 = 14660 nM T99799 CN4S6W 127025340 IC50 = 13490 nM T99799 C35YFW 127025347 IC50 = 14070 nM T99799 CU5Y2J 127025348 IC50 = 12440 nM T99799 CZNG40 127025349 IC50 = 11870 nM T99799 CQ32HN 127025350 IC50 = 14950 nM T99799 C8HT6M 127025617 IC50 = 2930 nM T99799 CH6A2X 127026192 IC50 = 1980 nM T99799 C2MHZ4 127026193 IC50 = 3450 nM T99799 C71BST 127026245 IC50 = 3800 nM T99799 C5NE2H 127027141 IC50 = 23790 nM T99799 CB25JK 127027142 IC50 = 26600 nM T99799 CT70GX 127027146 IC50 = 6120 nM T99799 CDV42T 127027424 IC50 = 14710 nM T99799 C6M5VF 127027425 IC50 = 15920 nM T99799 CX4YN3 127027643 IC50 = 15.7 nM T99799 C4AE0D 127027644 IC50 = 4.68 nM T99799 CJU4L1 127027645 IC50 = 10.8 nM T99799 CJWO49 127027646 IC50 = 80.6 nM T99799 CD5G9O 127027963 IC50 = 10.2 nM T99799 CBC0Y6 127028241 IC50 = 9000 nM T99799 C6R4EA 127028375 IC50 = 15090 nM T99799 CV5C7L 127028376 IC50 = 26130 nM T99799 C0NC1G 127028377 IC50 = 25420 nM T99799 CTF47Q 127028378 IC50 = 23810 nM T99799 CCO6D4 127028379 IC50 = 26040 nM T99799 C3DGN9 127029030 IC50 = 4900 nM T99799 C3FHL4 127029354 IC50 = 9100 nM T99799 CWJ80N 127029355 IC50 = 40000 nM T99799 C9RD5O 127029356 IC50 = 19300 nM T99799 C3BOU8 127029357 IC50 = 5700 nM T99799 C1QL4R 127033914 IC50 = 13 nM T99799 CF3HK1 127034304 IC50 > 200000 nM T99799 CY1I9K 127034570 IC50 = 163800 nM T99799 CZ3EV8 127035309 IC50 = 1.23 nM T99799 C7TQI5 127035310 IC50 = 8.89 nM T99799 C4HJR5 127036051 IC50 = 30 nM T99799 CKUR62 127036052 IC50 = 6.9 nM T99799 C1XE2Y 127036053 IC50 = 11.6 nM T99799 CF19QE 127036054 IC50 = 26.1 nM T99799 C07GWU 127036055 IC50 = 7.35 nM T99799 CA3MW8 127036212 IC50 = 31.9 nM T99799 COZ7S8 127036213 IC50 = 2.48 nM T99799 CW5MQ7 127036214 IC50 = 1.3 nM T99799 CPY5X2 127036215 IC50 = 0.49 nM T99799 C4JFN8 127036216 IC50 = 2.54 nM T99799 CX85YQ 127036232 IC50 = 2.3 nM T99799 CS6ND0 127036233 IC50 = 0.48 nM T99799 CVO6Y9 127036234 IC50 = 2.35 nM T99799 C1WLH2 127036472 IC50 = 30.9 nM T99799 C59WQJ 127036580 IC50 = 33.33 ug.mL-1 T99799 CM73TG 127036581 IC50 > 80 ug.mL-1 T99799 C65EVQ 127036864 IC50 = 8100 nM T99799 C0RXJ6 127036990 IC50 = 7900 nM T99799 C2LH5V 127037240 IC50 = 12.8 nM T99799 CH63BP 127037241 IC50 = 6.86 nM T99799 CIHE05 127037242 IC50 = 17.9 nM T99799 CG02IX 127037256 IC50 > 80 ug.mL-1 T99799 CMI6G3 127037257 IC50 = 66.67 ug.mL-1 T99799 C8S5LU 127037259 IC50 > 80 ug.mL-1 T99799 C8AYT1 127037384 IC50 = 4.87 nM T99799 C49PET 127037401 IC50 = 77 ug.mL-1 T99799 CUYD86 127037417 IC50 = 39.6 ug.mL-1 T99799 C3SN7K 127037516 IC50 > 80 ug.mL-1 T99799 CD16UI 127037518 IC50 > 80 ug.mL-1 T99799 CHR89X 127037869 IC50 = 16840 nM T99799 C0RTX1 127038878 IC50 = 24670 nM T99799 CO81HM 127038907 IC50 = 23770 nM T99799 C4QWS0 127043654 IC50 = 1030000 nM T99799 CQZW98 127043697 IC50 = 0.28 nM T99799 CCGN43 127043698 IC50 = 0.53 nM T99799 C7XP8D 127043699 IC50 = 1.17 nM T99799 CCRX05 127043700 IC50 = 42.7 nM T99799 C5IQU4 127043705 IC50 = 78.2 nM T99799 C09KSX 127043865 IC50 = 32.1 nM T99799 CG3DR4 127043866 IC50 = 2.85 nM T99799 CCWJ60 127043867 IC50 = 1.23 nM T99799 CG20QN 127043868 IC50 = 0.79 nM T99799 C3W8MB 127043871 IC50 = 15.9 nM T99799 C9M0KG 127043877 IC50 = 1230 nM T99799 CZA3R7 127043878 IC50 = 15.2 nM T99799 CX1G8L 127043879 IC50 = 122000 nM T99799 C54WIK 127043880 IC50 = 71.2 nM T99799 CP72LZ 127044176 IC50 = 0.27 nM T99799 C2VJ7H 127044293 IC50 = 400000 nM T99799 CF9BD1 127044471 IC50 = 1190000 nM T99799 C5GVQ3 127044472 IC50 = 800000 nM T99799 CT6YL4 127044473 IC50 = 400000 nM T99799 C7S5KZ 127044474 IC50 = 310000 nM T99799 CXS8Z2 127044620 IC50 = 900000 nM T99799 CS0CG7 127044621 IC50 = 8100 nM T99799 CI21OB 127044622 IC50 = 2000 nM T99799 C3PB5G 127044623 IC50 = 590 nM T99799 CXN83I 127044654 IC50 = 2.06 nM T99799 C97PFW 127044655 IC50 = 1.3 nM T99799 CC7W8O 127044656 IC50 = 1.15 nM T99799 C19MEI 127044657 IC50 = 3.51 nM T99799 CMU0Q3 127045144 IC50 = 1.44 nM T99799 CZOJ81 127045292 IC50 = 2.75 nM T99799 C37IKG 127045293 IC50 = 1.19 nM T99799 C8V2DN 127048404 IC50 = 1440 nM T99799 CQ16RS 127048405 IC50 = 669 nM T99799 CY71LG 127048406 IC50 = 7510 nM T99799 CW2B3M 127048716 IC50 = 784 nM T99799 CKEN30 127048749 IC50 = 1220 nM T99799 C23EOB 127049071 IC50 = 690 nM T99799 CU8I7J 127049072 IC50 = 988 nM T99799 C23YAL 127049073 IC50 = 245 nM T99799 C2BVI5 127049123 IC50 = 850 nM T99799 CG65ES 127049124 IC50 = 1400 nM T99799 CR39WO 127049125 IC50 = 290 nM T99799 C7X0IE 127049126 IC50 = 1060 nM T99799 CU85GC 127049730 IC50 = 76 nM T99799 CRW64G 127049731 IC50 = 3240 nM T99799 CXB9K4 127050511 IC50 = 950 nM T99799 CCI4E1 127050512 IC50 = 1420 nM T99799 CZGX21 127050513 IC50 = 1030 nM T99799 CS8X7B 127050845 IC50 = 2210 nM T99799 CRE9O5 127051536 IC50 = 286 nM T99799 C39VRD 127051623 IC50 = 400 nM T99799 C5CYS7 127051624 IC50 = 3010 nM T99799 CN63WP 129766223 IC50 = 520 nM T99799 CYQT64 129904916 IC50 > 100000 nM T99799 C3OH2U 132281442 IC50 = 68.2 nM T99799 CZ2JQ4 132427688 IC50 = 260 nM T99799 C61DGH 132495293 IC50 = 1020 nM T99799 C5AU1H 132495295 IC50 = 5270 nM T99799 CZ3OD0 132495360 IC50 = 2600 nM T99799 CBN5C0 132495361 IC50 = 127 nM T99799 CM7PY1 132547201 Ki = 160 nM T99799 C3F4ME 132569621 IC50 = 7300 nM T99799 CX59ME 133561407 IC50 > 10000 nM T99799 C4YH6G 134129916 IC50 = 25400 nM T99799 C0EU7L 134130629 IC50 = 6350 nM T99799 C5Z9WG 134131252 IC50 = 29.7 nM T99799 C8R7KL 134131932 IC50 = 52.44 nM T99799 CCJF74 134132255 IC50 = 39 nM T99799 C3VO0S 134132482 IC50 = 8 nM T99799 C9UGN0 134132984 IC50 = 37 nM T99799 CA5BJ4 134133150 IC50 = 6.4 nM T99799 C6VS5U 134133379 IC50 = 137 nM T99799 CVF3T5 134133384 IC50 = 30 nM T99799 CZTV48 134134429 IC50 = 4370 nM T99799 CYB1T5 134134557 IC50 = 30.41 nM T99799 CB31IT 134134606 IC50 = 8550 nM T99799 CYWV57 134134625 IC50 > 10000 nM T99799 C71IYO 134135593 IC50 = 15 nM T99799 CP1E5Y 134135669 IC50 = 3.79 nM T99799 CB19DO 134135810 IC50 = 65 nM T99799 CZ9YA3 134135893 IC50 = 7360 nM T99799 C9OE5Y 134135942 IC50 = 760 nM T99799 C8X1DP 134136230 IC50 = 5 nM T99799 CHB06R 134136355 IC50 = 41400 nM T99799 CP3RN6 134136543 IC50 = 1020 nM T99799 CK06MI 134136825 IC50 = 49200 nM T99799 CM83OH 134137000 IC50 = 1910 nM T99799 C7XE0G 134137541 IC50 = 5120 nM T99799 CSA09I 134137557 IC50 = 79 nM T99799 C97CUD 134137716 IC50 = 64 nM T99799 CYG95X 134137746 IC50 = 18800 nM T99799 C9JW0A 134137761 IC50 = 6080 nM T99799 CZB2H1 134137882 IC50 = 73 nM T99799 C3MFB4 134138158 IC50 = 3.59 nM T99799 C3WL0X 134138347 IC50 = 5600 nM T99799 CTQY30 134138725 IC50 = 37400 nM T99799 C5B6YK 134138931 IC50 = 43 nM T99799 CYR2D1 134138980 IC50 = 48.13 nM T99799 CQU8T5 134139124 IC50 = 281 nM T99799 C32PAF 134139263 IC50 > 200000 nM T99799 C6BH1E 134139570 IC50 = 12 nM T99799 CM5D2F 134139579 IC50 = 65700 nM T99799 C5E6PV 134139682 IC50 = 42 nM T99799 C0VGT1 134140048 IC50 = 5000 nM T99799 COB3U4 134140335 IC50 = 4370 nM T99799 C1A7EP 134140534 IC50 = 570 nM T99799 CBS53R 134140571 IC50 = 4.12 nM T99799 CH2W1P 134140732 IC50 = 6 nM T99799 C73LGF 134140781 IC50 = 8641 nM T99799 CU2H9S 134140801 IC50 = 6.97 nM T99799 CYW3P5 134141480 IC50 = 53.76 nM T99799 C6NCM8 134141704 IC50 = 10 nM T99799 CC6P0J 134141898 IC50 = 38900 nM T99799 CHDC50 134142324 IC50 = 15 nM T99799 CSYM31 134142478 IC50 = 23444 nM T99799 CUP09Q 134142596 IC50 = 4390 nM T99799 C9L1VS 134142725 IC50 = 1560 nM T99799 CI38NM 134143999 IC50 = 2870 nM T99799 C47KWL 134144584 IC50 = 4040 nM T99799 CIE6T7 134144753 IC50 = 21 nM T99799 CZ4WL3 134144932 IC50 = 365 nM T99799 CKAF58 134145123 IC50 = 15 nM T99799 C4Z9HA 134145445 IC50 = 30 nM T99799 CP0D4F 134146126 IC50 = 1223 nM T99799 CZVL70 134146128 IC50 = 12800 nM T99799 C89RCM 134146339 IC50 = 78700 nM T99799 C1K2XO 134146719 IC50 = 2520 nM T99799 CZM9O4 134146757 IC50 = 5890 nM T99799 CBOY65 134146798 IC50 = 24 nM T99799 CW1U8M 134147085 IC50 = 3370 nM T99799 CID47M 134147264 IC50 = 7 nM T99799 C3G2FL 134147416 IC50 = 47.33 nM T99799 CNVG70 134147548 IC50 > 10000 nM T99799 C5A1SG 134147628 IC50 = 1420 nM T99799 C5E6RH 134147648 IC50 > 10000 nM T99799 CE7X9I 134148653 IC50 = 7 nM T99799 CXOD70 134148863 IC50 = 32.07 nM T99799 C7E3YA 134149382 IC50 > 10000 nM T99799 C03PFN 134149524 IC50 = 3930 nM T99799 CSMP25 134149784 IC50 = 3060 nM T99799 C4Y5ZX 134150471 IC50 = 260 nM T99799 CRZ2W4 134150858 IC50 = 3306 nM T99799 C5BMP0 134151164 IC50 = 456.21 nM T99799 C4RD1Z 134151725 IC50 = 22.56 nM T99799 CJ98WY 134152913 IC50 = 6400 nM T99799 CIV53R 134153098 IC50 = 11.58 nM T99799 CE0DW1 134153138 IC50 = 4480 nM T99799 CA2KR0 134153338 IC50 = 2 nM T99799 CT51CQ 134153533 IC50 = 13 nM T99799 CPBG73 134153558 IC50 = 4590 nM T99799 CNC58Z 134154903 IC50 = 9 nM T99799 CO8IQ0 134155051 IC50 = 1.8 nM T99799 C9QXG2 134155279 IC50 = 23 nM T99799 CA59GH 134155309 IC50 = 75 nM T99799 CJ7Y1Q 134155675 IC50 = 50200 nM T99799 CQA14Y 134155772 IC50 = 384 nM T99799 CL80HA 134155833 IC50 = 13 nM T99799 CPBJ79 134155988 IC50 = 76900 nM T99799 CS3X9K 134156217 IC50 = 29 nM T99799 CC84RT 134157228 IC50 = 2190 nM T99799 CC0IG7 134157232 IC50 = 54396 nM T99799 CW4H7K 134157259 IC50 = 8 nM T99799 CT0IZ2 134157388 IC50 = 77 nM T99799 CY65KP 134157669 IC50 = 11 nM T99799 CJS28R 134157781 IC50 = 18 nM T99799 CUD08L 134817200 IC50 = 1690 nM T99799 CEW6B4 135401162 IC50 = 4000 nM T99799 CQ0WB8 135409581 IC50 > 50000 nM T99799 CXS6M1 135410029 Ki = 390000 nM T99799 C6SMT5 135517369 IC50 = 2200 nM T99799 C5ZCK6 135531254 IC50 > 50000 nM T99799 C8TQ1R 135595416 IC50 = 16000 nM T99799 C73ZKR 135599085 IC50 = 2500 nM T99799 C5YH3F 135621406 IC50 = 194 nM T99799 CFNX32 135777608 Ki = 212400 nM T99799 C98KNJ 135846078 IC50 > 10000 nM T99799 C81ITK 135846093 IC50 > 10000 nM T99799 C8I1WV 135905682 IC50 = 14000 nM T99799 CC2L8T 136044207 IC50 = 13700 nM T99799 CQSW91 136110931 IC50 = 140220 nM T99799 CB1ZV3 136110932 IC50 = 101520 nM T99799 CZ8UM3 136239360 IC50 = 3310 nM T99799 C4TR7Z 136239361 IC50 = 57810 nM T99799 CW2NC0 136239465 Ki = 446480 nM T99799 C92YAW 136239487 IC50 = 231610 nM T99799 CO1TR8 136242439 IC50 = 23000 nM T99799 CL0W4D 136244480 IC50 = 58250 nM T99799 CW4LE8 136244481 IC50 = 358 nM T99799 CKCE30 136244497 IC50 = 8810 nM T99799 CU5VF2 136244586 IC50 = 56810 nM T99799 CV3ST2 136254438 IC50 = 38510 nM T99799 CNG5M3 136254439 IC50 = 75410 nM T99799 CH29ZJ 136254440 IC50 = 8110 nM T99799 CYD96O 136254441 IC50 = 116610 nM T99799 C86MBG 136260466 IC50 = 136910 nM T99799 CKC84W 136260526 IC50 = 57110 nM T99799 CVE2S8 136260527 IC50 = 68410 nM T99799 C1X8GA 136260528 IC50 = 56510 nM T99799 CJZ38F 136264303 IC50 = 64320 nM T99799 C7CGQ4 136264469 IC50 = 52140 nM T99799 COQ2J8 136264470 IC50 = 19370 nM T99799 C5CB7E 136268789 IC50 > 50000 nM T99799 CEBX51 136498868 IC50 = 3970 nM T99799 CYM59N 136498869 IC50 = 4700 nM T99799 C8BAP5 137125243 IC50 = 24100 nM T99799 C8T1NA 137169079 IC50 > 50000 nM T99799 CEL8Q2 137631614 IC50 = 4780 nM T99799 CRH92A 137632694 IC50 = 18 nM T99799 CX6YO4 137632785 IC50 > 5000 nM T99799 CG21YK 137632803 IC50 = 20020 nM T99799 CIY0P1 137632867 IC50 = 400 nM T99799 CQE2C5 137633051 IC50 = 300 nM T99799 C8FSZ4 137633176 IC50 > 5000 nM T99799 CC3Z7H 137633188 IC50 = 40950 nM T99799 C0Y2FZ 137633400 IC50 = 9910 nM T99799 CVK1Z4 137633425 IC50 = 22150 nM T99799 C02GNF 137633542 IC50 = 410 nM T99799 CEI0T6 137633782 IC50 = 14600 nM T99799 C9QLT1 137633879 IC50 = 5690 nM T99799 CCF19I 137634197 IC50 = 50 nM T99799 CVK63S 137634258 IC50 = 3500 nM T99799 C0T9ZD 137634437 IC50 = 3830 nM T99799 CXDY28 137634711 IC50 > 50000 nM T99799 CUSI50 137634757 IC50 > 5000 nM T99799 CH2IJ8 137634974 IC50 = 9100 nM T99799 CU0DK7 137635136 IC50 = 9800 nM T99799 CJ21RK 137635381 IC50 = 390 nM T99799 C7S9TN 137635450 IC50 = 1100 nM T99799 CF08CP 137635497 IC50 = 376710 nM T99799 CK12JV 137635625 IC50 = 230 nM T99799 C82ELC 137635812 IC50 = 82000 nM T99799 C1GT8Y 137635839 IC50 = 302450 nM T99799 C9GA2C 137635913 IC50 = 1584.89 nM T99799 CWSF64 137636375 IC50 = 54100 nM T99799 CV8W7S 137637059 IC50 > 50000 nM T99799 C2WBP4 137637064 IC50 = 3200 nM T99799 C2Z5KH 137637592 IC50 = 6720 nM T99799 CZ5WE1 137637732 IC50 > 50000 nM T99799 CWB7O3 137637856 IC50 = 55 nM T99799 CFP1G9 137637896 IC50 = 11460 nM T99799 CFI74R 137637910 IC50 = 3600 nM T99799 C07FMS 137638163 IC50 > 5000 nM T99799 CC7E4I 137638765 IC50 > 50000 nM T99799 CR5G9J 137638769 IC50 = 1600 nM T99799 CJP8W9 137638885 IC50 = 74250 nM T99799 C4AX5H 137639047 IC50 = 12900 nM T99799 C6DJ8C 137639617 IC50 = 2230 nM T99799 C89ELW 137639718 IC50 = 10200 nM T99799 CRG16O 137639776 IC50 = 11380 nM T99799 CJ1L2M 137639795 IC50 = 150 nM T99799 CPK5O7 137639919 IC50 > 5000 nM T99799 C7EN5K 137640663 IC50 = 10100 nM T99799 CLS48N 137641195 IC50 = 97000 nM T99799 CJ1V3P 137641233 IC50 = 4840 nM T99799 CY5NR3 137641257 IC50 > 50000 nM T99799 CTR8E0 137641522 IC50 = 5011.87 nM T99799 CXL6G5 137641793 IC50 = 8470 nM T99799 CED9V8 137641985 IC50 = 1700 nM T99799 CDY1X7 137641989 IC50 = 20580 nM T99799 CH8B5Q 137642077 IC50 = 7140 nM T99799 C3EL4I 137642431 IC50 = 5600 nM T99799 C6BZ2P 137642547 IC50 = 5490 nM T99799 CH2A8I 137642953 IC50 = 11670 nM T99799 CT72VS 137643173 IC50 > 5000 nM T99799 C15JOE 137643788 IC50 = 5900 nM T99799 C49CZB 137643848 IC50 > 5000 nM T99799 C9B2ZE 137644072 IC50 = 71000 nM T99799 CM2CG5 137644485 IC50 = 286720 nM T99799 C5OEB2 137644607 IC50 > 5000 nM T99799 C4YGM1 137644680 IC50 > 5000 nM T99799 CM91SH 137644867 IC50 = 13050 nM T99799 C7TWP1 137644997 IC50 = 8900 nM T99799 CSCI58 137645198 IC50 = 10410 nM T99799 C1DHM4 137645326 IC50 = 8200 nM T99799 CG96IN 137645336 IC50 = 5710 nM T99799 CAOM59 137645444 IC50 = 12970 nM T99799 C4OQ9U 137645703 IC50 = 6100 nM T99799 CC2SY8 137646193 IC50 > 50000 nM T99799 CPV4Z7 137646357 IC50 = 25900 nM T99799 C5CPS2 137646394 Ki = 0.0111 nM T99799 CAGB15 137646401 IC50 = 3800 nM T99799 CV0I6J 137647059 IC50 = 14190 nM T99799 CL45YE 137647453 IC50 = 2990 nM T99799 C9J3XC 137647729 IC50 = 5000 nM T99799 CO3P1M 137647800 IC50 = 22680 nM T99799 CNUC94 137647812 IC50 = 110000 nM T99799 C5MJG7 137647822 IC50 = 1000 nM T99799 C0ZXC8 137647877 IC50 = 300 nM T99799 C41KDG 137648030 IC50 > 50000 nM T99799 CEC78J 137648049 IC50 = 70 nM T99799 CJP1G6 137648183 IC50 = 30400 nM T99799 CC5R7U 137648202 IC50 = 9600 nM T99799 CBPK31 137648694 IC50 = 2511.89 nM T99799 C07ZJU 137648924 IC50 = 16880 nM T99799 CMRI71 137649149 IC50 = 2300 nM T99799 CW2UK0 137649211 IC50 = 8600 nM T99799 C30VHY 137649676 IC50 = 145690 nM T99799 C6JEQ0 137649792 IC50 = 1350 nM T99799 C7Z4MI 137649813 IC50 = 14000 nM T99799 C12HUM 137650006 IC50 = 25000 nM T99799 CBFM14 137650067 IC50 > 10000 nM T99799 C0ZM5Q 137650571 IC50 = 632 nM T99799 CH50RP 137650702 IC50 = 1200 nM T99799 CHW83L 137650736 IC50 = 67 nM T99799 CJW29P 137650881 IC50 = 3800 nM T99799 C54VBE 137651033 IC50 = 2760 nM T99799 CTOX45 137651149 IC50 = 1437 nM T99799 CXM65D 137651291 IC50 = 110000 nM T99799 CWQ87J 137651676 IC50 = 702 nM T99799 C3WL9S 137652298 IC50 = 1850 nM T99799 CW9HL2 137652394 IC50 = 360 nM T99799 C1KSJ8 137652783 IC50 = 4780 nM T99799 CHWO15 137652896 IC50 = 7800 nM T99799 CMP3S2 137652915 IC50 = 1560 nM T99799 CQJ78X 137653099 IC50 = 4860 nM T99799 CFPV35 137653376 IC50 = 2340 nM T99799 CSO97E 137653574 IC50 = 4500 nM T99799 CG3V4T 137653648 IC50 = 1200 nM T99799 C6O0AJ 137653712 IC50 = 9700 nM T99799 CX4AM2 137653862 IC50 = 5760 nM T99799 CB1I0V 137654237 IC50 = 23280 nM T99799 C0UNA5 137654399 IC50 = 9500 nM T99799 C0C5OB 137654571 IC50 = 50118.72 nM T99799 C0LR3F 137654627 IC50 > 50000 nM T99799 CO25BH 137654740 IC50 > 5000 nM T99799 CT1PA9 137654741 IC50 = 1300 nM T99799 C58UJM 137654765 IC50 = 41760 nM T99799 C4UZ6L 137654824 IC50 = 7.28 nM T99799 CAQ92O 137654935 IC50 > 5000 nM T99799 CP3R6K 137655004 IC50 = 8900 nM T99799 CS7G0V 137655713 IC50 = 3100 nM T99799 CCA96J 137655921 IC50 = 2200 nM T99799 CMA9P4 137655981 IC50 > 50000 nM T99799 C4XM2Y 137657255 IC50 > 5000 nM T99799 CA26MD 137657287 IC50 = 2500 nM T99799 C61BAH 137657694 IC50 = 25070 nM T99799 CJNL70 137657810 IC50 = 3980 nM T99799 C9XPC4 137657910 IC50 = 17600 nM T99799 CU4B0Q 137658210 IC50 = 170 nM T99799 CT51VW 137658213 IC50 = 24900 nM T99799 CN0SF1 137658402 IC50 = 2140 nM T99799 CW2I9D 137658492 IC50 = 3630 nM T99799 C15GDM 137658514 IC50 = 12080 nM T99799 CQC6G7 137658542 IC50 = 5700 nM T99799 CJU20M 137658706 IC50 = 1300 nM T99799 CC7V1S 137658749 IC50 = 5450 nM T99799 CEV12H 137659101 IC50 = 8800 nM T99799 COL58K 137659202 IC50 = 29800 nM T99799 CSP06U 137659306 IC50 = 29800 nM T99799 CC65MS 137659483 IC50 = 30500 nM T99799 CBD24K 137660365 IC50 = 15800 nM T99799 C8IW5O 137660695 IC50 > 5000 nM T99799 CH34LO 137660979 IC50 = 4030 nM T99799 CKMC76 137661029 IC50 = 12680 nM T99799 C6F7QS 137661135 IC50 = 7.12 nM T99799 C31MDX 137661164 IC50 > 50000 nM T99799 C7E2OH 137661175 IC50 > 5000 nM T99799 CD8W3T 137661581 IC50 = 38.24 nM T99799 C7FL2W 137661647 IC50 = 8400 nM T99799 CQV79Z 137661668 IC50 > 50000 nM T99799 CIJ43L 137662097 IC50 = 263110 nM T99799 C9J4DH 138320049 IC50 = 254 nM T99799 CU3VY8 141700626 IC50 = 2100 nM T99799 CY20TH 141700627 IC50 = 0.26 nM T99799 CC50YG 141700631 IC50 = 230 nM T99799 CU7SJ0 145722355 IC50 = 2.5 nM T99799 C80HQW 145949396 IC50 = 5680 nM T99799 CZ0IR5 145949784 IC50 = 1560 nM T99799 CU15AO 145950308 IC50 = 8410 nM T99799 C3GNZ9 145950384 IC50 = 511 nM T99799 CFU46Z 145950418 IC50 = 310 nM T99799 CN1MF4 145950493 IC50 = 3190 nM T99799 C35CUT 145950652 IC50 = 1270 nM T99799 CQWI16 145950841 IC50 = 356 nM T99799 CN4C6I 145951178 IC50 > 10000 nM T99799 C81CRX 145951391 IC50 = 5270 nM T99799 CSU4Y2 145951896 IC50 = 6540 nM T99799 CL1TK4 145952378 IC50 = 47210 nM T99799 CR26YA 145952393 IC50 = 630 nM T99799 C6VLZ8 145952662 IC50 = 3690 nM T99799 CY7RD4 145953155 IC50 = 378 nM T99799 C2SFL4 145953212 IC50 = 37500 nM T99799 C5U8LK 145953230 IC50 = 4020 nM T99799 C9ZPF5 145954333 IC50 = 372 nM T99799 CP8L3U 145954454 IC50 = 452 nM T99799 CB2PU4 145954736 IC50 = 340 nM T99799 C8LJV7 145954769 IC50 = 1110 nM T99799 CF09RS 145954786 IC50 = 510 nM T99799 CRP68J 145955177 IC50 = 2650 nM T99799 CMYF60 145956446 IC50 = 11700 nM T99799 CRTG06 145956559 IC50 = 3470 nM T99799 CNIR29 145956699 IC50 = 4010 nM T99799 C0Q3MP 145957027 IC50 = 650 nM T99799 C7BY3Q 145957085 IC50 = 2680 nM T99799 COR92I 145957306 IC50 = 9960 nM T99799 CW1M4Y 145958077 IC50 = 4590 nM T99799 C7UK4Q 145958135 IC50 = 990 nM T99799 CG6D8I 145958306 IC50 > 10000 nM T99799 CCBO90 145958532 IC50 > 10000 nM T99799 CTCE08 145958953 IC50 = 25800 nM T99799 C7E0WG 145959287 IC50 = 828 nM T99799 CNS69M 145959783 IC50 > 10000 nM T99799 CLP6E5 145959857 IC50 = 14930 nM T99799 CFUJ38 145959883 IC50 = 10000 nM T99799 CRD76Q 145963428 IC50 = 32530 nM T99799 CD6K7P 145963526 IC50 = 4700 nM T99799 C37BNF 145963787 IC50 = 37.2 nM T99799 CTH70Y 145963788 IC50 = 8320 nM T99799 C85ZOK 145963821 IC50 = 1320 nM T99799 C8VFP2 145963831 IC50 = 20.7 nM T99799 CIZ2D6 145964146 IC50 = 408 nM T99799 CUY37P 145964192 IC50 = 1186 nM T99799 CL8IM7 145964214 IC50 = 3340 nM T99799 CCX4G7 145964403 IC50 = 16.6 nM T99799 C7O1VM 145964717 IC50 = 1001 nM T99799 CC65HS 145965070 IC50 = 12.4 nM T99799 C52IFK 145965199 IC50 = 577 nM T99799 CO09TS 145966146 IC50 = 107 nM T99799 CZ20XJ 145967112 IC50 = 12400 nM T99799 CCVM34 145967131 IC50 = 3720 nM T99799 C4RFE9 145967436 IC50 = 2400 nM T99799 C4CGL8 145968916 IC50 = 4.35 nM T99799 C7NB8L 145970781 IC50 = 103 nM T99799 C8IRS3 145970790 IC50 = 4950 nM T99799 CNS36B 145971232 IC50 = 1750 nM T99799 CS52IM 145971379 IC50 = 48.8 nM T99799 CS2NH6 145971450 IC50 = 154000 nM T99799 CKP39X 145971650 IC50 = 1080 nM T99799 C0RV3Z 145972056 IC50 = 1190 nM T99799 C10KGM 145972388 IC50 = 1030 nM T99799 CADI36 145972622 IC50 = 1290 nM T99799 CVG37T 145972858 IC50 = 26.8 nM T99799 CC3K4N 145972893 IC50 = 8860 nM T99799 CMB59C 145972994 IC50 = 1460 nM T99799 CHA90Q 145973001 IC50 = 145 nM T99799 CE9U6I 145973015 IC50 = 83.3 nM T99799 C8X5YT 145973525 IC50 = 8010 nM T99799 CR01XP 145973666 IC50 = 674 nM T99799 CV2I6R 145973676 IC50 = 950 nM T99799 CP3W4L 145974148 IC50 = 3120 nM T99799 C7WRK1 145974265 IC50 = 7740 nM T99799 CUD2Z0 145974298 IC50 = 45500 nM T99799 C9KNC3 145974491 IC50 = 13400 nM T99799 C2CSU4 145974513 IC50 = 10.5 nM T99799 C8VZ5F 145974561 IC50 > 10000 nM T99799 CJ51HA 145974740 IC50 = 81.5 nM T99799 C5UZ8W 145974825 IC50 = 507 nM T99799 CXS48G 145974962 IC50 = 49300 nM T99799 C80VLM 145975022 IC50 = 107 nM T99799 C26ZBO 145975126 IC50 = 6160 nM T99799 CU2ES3 145975561 IC50 = 45.7 nM T99799 CU1NO6 145976650 IC50 = 280 nM T99799 CEXP52 145976876 IC50 = 16600 nM T99799 CRAM60 145977029 IC50 = 1050 nM T99799 CF4A0B 145977178 IC50 = 2.35 nM T99799 CBFC12 145977206 IC50 = 2030 nM T99799 CEO72I 145977249 IC50 = 29.9 nM T99799 COSM78 145977433 IC50 = 16.3 nM T99799 CL9HU4 145977623 IC50 = 108 nM T99799 CKO6P0 145977734 IC50 = 4320 nM T99799 C2UVJ5 145977785 IC50 = 1210 nM T99799 CYW3U1 145978073 IC50 = 58.9 nM T99799 CUD60Z 145978446 IC50 = 823 nM T99799 CQ6TB5 145978697 IC50 = 37200 nM T99799 CE07DW 145978744 IC50 = 1280 nM T99799 CHX28E 145978908 IC50 = 10300 nM T99799 CZG8R6 145979011 IC50 = 210 nM T99799 C9RQ7P 145979084 IC50 = 670 nM T99799 CXD4H1 145979225 IC50 = 6916.4 nM T99799 CJYX43 145979238 IC50 = 9.5 nM T99799 CGWB38 145979348 Ki = 187000 nM T99799 C7XLF0 145979801 IC50 = 4.571 nM T99799 CX2RW9 145979866 IC50 = 19560 nM T99799 C1D9ZU 145979972 IC50 > 10000 nM T99799 CE0DG7 145980262 IC50 = 265.8 nM T99799 C6PL4V 145980390 IC50 = 1949.84 nM T99799 CW93VH 145980588 IC50 > 10000 nM T99799 CK59PS 145980980 IC50 = 237 nM T99799 CSNL80 145981760 IC50 = 21.8 nM T99799 C8TP1V 145981823 IC50 > 10000 nM T99799 CE84KA 145981976 Ki = 195000 nM T99799 CX3M9J 145981988 IC50 = 4440 nM T99799 CLD9H6 145982286 IC50 = 28 nM T99799 CWNB08 145982383 IC50 = 4250 nM T99799 CFNJ87 145982457 IC50 = 9300 nM T99799 C7VJ1L 145983695 IC50 = 23600 nM T99799 C53SFP 145984170 IC50 = 634.5 nM T99799 CW4X2T 145984359 IC50 > 10000 nM T99799 CSYF87 145984930 IC50 = 103.1 nM T99799 C19IWK 145986527 IC50 = 450 nM T99799 CD73AY 145986601 IC50 = 8790 nM T99799 CCWA30 145986676 IC50 = 20000 nM T99799 CS1CL3 145986706 IC50 = 200 nM T99799 CGLW18 145987198 Ki = 273000 nM T99799 CBG81P 145987259 Ki = 294000 nM T99799 C21BYI 145987407 IC50 = 4300 nM T99799 CAXH94 145987711 IC50 = 28 nM T99799 CJP7H5 145987783 IC50 = 100 nM T99799 C98DHT 145987800 IC50 > 10000 nM T99799 CA82TF 145987838 IC50 = 5800 nM T99799 CLGS98 145988032 IC50 > 10000 nM T99799 C3M1ZO 145988042 IC50 > 10000 nM T99799 CA45JZ 145988111 IC50 = 263.03 nM T99799 C1XU7P 145988798 IC50 > 10000 nM T99799 C2A8MY 145989254 IC50 = 39300 nM T99799 CLG23Y 145989395 IC50 = 20951.3 nM T99799 C6RB3V 145989629 IC50 > 10000 nM T99799 C5BFR8 145989798 IC50 = 19 nM T99799 C6QRA9 145989946 IC50 = 7420 nM T99799 C4OAU8 145989956 IC50 > 10000 nM T99799 CVBP12 145989988 IC50 > 10000 nM T99799 C9NTF8 145990243 IC50 > 10000 nM T99799 C63USF 145990366 Ki = 265000 nM T99799 CDBW68 145990442 IC50 = 9610 nM T99799 C4N1WB 145990478 IC50 = 1.82 nM T99799 CGP60E 145990565 IC50 = 6300 nM T99799 CR59TZ 145990611 IC50 = 9900 nM T99799 CQ4R9F 145990749 IC50 = 84810 nM T99799 CCAM14 145990761 IC50 = 74240 nM T99799 C5QZJ4 145990784 IC50 > 10000 nM T99799 C6AZ2B 145990932 IC50 = 228.6 nM T99799 CK9Z4O 145991455 IC50 = 135 nM T99799 CKQ9N2 145991501 IC50 = 11300 nM T99799 C1ZQ0W 145991508 IC50 = 1570 nM T99799 CQD5J2 145991584 IC50 = 460.4 nM T99799 C1P4MD 145991603 IC50 = 48.1 nM T99799 C8KUE6 145991747 IC50 = 610 nM T99799 CR69KG 145992024 IC50 = 51 nM T99799 C1O3VK 145992136 IC50 = 9310 nM T99799 C84LNF 145992210 Ki = 140000 nM T99799 CB9P8D 145992212 IC50 > 10000 nM T99799 C1WI3A 145992723 IC50 > 10000 nM T99799 C7WA5I 145992788 IC50 = 9 nM T99799 CPBJ68 145992936 IC50 > 10000 nM T99799 CF36AC 145993120 IC50 = 5090 nM T99799 CBK49L 145993204 IC50 = 71 nM T99799 C1FBD7 145993205 IC50 = 150 nM T99799 C5YMR4 145993208 IC50 = 6500 nM T99799 CI9T7A 145993228 IC50 = 1611.8 nM T99799 CNDI85 145993235 IC50 = 2485.1 nM T99799 CQ61NL 145993296 IC50 = 7823 nM T99799 CY2N1D 145993326 IC50 = 4320 nM T99799 CUVC73 145993378 IC50 > 10000 nM T99799 CK54FE 145993438 IC50 > 10000 nM T99799 C30CMY 145993498 IC50 > 10000 nM T99799 C27FDC 145993580 IC50 > 10000 nM T99799 CQ9HB3 145993722 IC50 = 2.29 nM T99799 CY62QA 145993943 Ki = 1.09 nM T99799 CQEN91 145993998 IC50 = 1794.2 nM T99799 C4V2RJ 145994271 IC50 = 9880 nM T99799 CC27PZ 146443282 IC50 = 2290 nM T99799 C06YAR 153979960 IC50 = 4000 nM T99799 CJ8V4Q 153979967 IC50 = 600 nM T99799 C5B1RI 153979968 IC50 = 1300 nM T99799 CZ2OW7 153979970 IC50 = 0.07 nM T99799 C2H9LT 153979972 IC50 = 70 nM T99799 CD6EF5 153979973 IC50 = 800 nM T99799 C15LBY 153979974 IC50 > 10000 nM T99799 CTV4G0 153979975 IC50 > 10000 nM T99799 CS4E3M 153979977 IC50 = 0.15 nM T99799 CH6A9F 153979986 IC50 = 9400 nM T99799 CBXN70 153979988 IC50 > 10000 nM T99799 C9L8CY 153979991 IC50 = 80 nM T99799 C94IGO 155510425 IC50 = 301 nM T99799 C0AZ2W 155510575 IC50 = 6030 nM T99799 CRX53K 155510902 IC50 = 426 nM T99799 C2TRD5 155511051 IC50 = 328 nM T99799 CH4PT0 155511056 IC50 > 50000 nM T99799 CQD8U1 155511223 IC50 = 6 nM T99799 C0TY4L 155512256 IC50 > 50000 nM T99799 C30QIL 155512277 IC50 > 50000 nM T99799 CYT0U1 155512533 IC50 = 933.25 nM T99799 CN1L2G 155512563 IC50 = 7060 nM T99799 C2OVJ6 155513058 IC50 > 50000 nM T99799 C8QOL4 155513096 IC50 = 40 nM T99799 CLP7Q5 155513372 IC50 = 2300 nM T99799 C8S4OV 155513382 IC50 > 10000 nM T99799 CQ4MT7 155514267 IC50 > 50000 nM T99799 CE31CI 155514453 IC50 = 2950 nM T99799 CY0E3D 155514519 IC50 = 11000 nM T99799 C4QTY1 155514573 IC50 = 25.6 nM T99799 C36OGK 155514733 IC50 > 50000 nM T99799 CBKQ23 155514904 IC50 = 41.69 nM T99799 CS0C1V 155515351 IC50 = 6.31 nM T99799 C8WO0D 155515901 IC50 = 11700 nM T99799 C37OWC 155516090 IC50 = 13400 nM T99799 CTR7C8 155516568 IC50 = 7220 nM T99799 COIQ70 155516605 IC50 = 67.8 nM T99799 CI02NB 155516607 IC50 = 395 nM T99799 CR4P3Z 155516698 IC50 = 3100 nM T99799 COQ0I2 155517103 IC50 = 8410 nM T99799 C7WQF6 155517133 IC50 = 38.9 nM T99799 C7CN4W 155517273 IC50 = 340 nM T99799 CFG9A1 155517376 IC50 = 54 nM T99799 C0DR8X 155517455 IC50 = 1020 nM T99799 CEU36W 155517463 IC50 > 50000 nM T99799 C62HKG 155518395 IC50 = 206 nM T99799 C0DUP5 155518577 IC50 = 27360 nM T99799 COR6Z3 155518726 IC50 = 65 nM T99799 CWA5P2 155518864 IC50 > 10000 nM T99799 CT5X0O 155519170 IC50 = 12.59 nM T99799 C0XI2C 155519241 IC50 = 48.2 nM T99799 CWOJ19 155519277 IC50 = 2740 nM T99799 CET82F 155519354 IC50 = 5300 nM T99799 CEJ87B 155519446 IC50 = 180 nM T99799 C1DVS3 155519968 IC50 = 125.3 nM T99799 CW65KH 155520207 IC50 = 140 nM T99799 CAIX71 155520508 IC50 > 10000 nM T99799 CZR0D3 155520717 IC50 = 5500 nM T99799 CHG5D0 155521756 IC50 = 7300 nM T99799 C9AT3Q 155521926 IC50 = 0.0017 nM T99799 CC2U3Z 155522419 IC50 = 1210 nM T99799 C2ML7G 155522745 IC50 = 9970 nM T99799 CF1OL6 155523160 IC50 = 4520 nM T99799 C1AEU5 155523624 IC50 = 48.98 nM T99799 C2ES7G 155523649 IC50 = 3900 nM T99799 CU0E6I 155523688 IC50 = 251.19 nM T99799 CS6IJ2 155524198 IC50 > 30000 nM T99799 C9VWZ8 155524523 IC50 = 79.43 nM T99799 CH24YB 155525250 IC50 = 398.11 nM T99799 CGMH43 155525252 IC50 = 64 nM T99799 C32XUD 155525503 IC50 = 190.55 nM T99799 CNB25L 155525773 IC50 > 100000 nM T99799 C3K9OH 155526042 IC50 = 13.18 nM T99799 CMT9X3 155526434 IC50 = 2.512 nM T99799 C6NU8X 155526479 IC50 = 56 nM T99799 CDY49N 155526514 IC50 = 501.19 nM T99799 CK85TG 155526796 IC50 = 123 nM T99799 CU0X9B 155526812 IC50 = 7.413 nM T99799 C9ZR4K 155526939 IC50 = 32.6 nM T99799 C68XKW 155527023 IC50 = 307 nM T99799 C1UOP6 155528201 IC50 = 4520 nM T99799 CR7VW0 155528538 IC50 > 10000 nM T99799 C68UIE 155528833 IC50 > 100000 nM T99799 CE98VB 155529070 IC50 = 2400 nM T99799 CC25TX 155530201 IC50 > 100000 nM T99799 CT80OY 155530802 IC50 = 158.49 nM T99799 C1V6BO 155531034 IC50 = 0.17 nM T99799 C2GH4F 155531521 IC50 = 3100 nM T99799 C3E5FM 155531627 IC50 = 140 nM T99799 CWB5N8 155532073 IC50 = 6420 nM T99799 C15PWD 155532152 IC50 = 36.1 nM T99799 C6XQF3 155532358 IC50 = 174 nM T99799 C3G4ZQ 155532469 IC50 = 970 nM T99799 CE13NX 155532485 IC50 = 32.36 nM T99799 CQL91M 155532503 IC50 = 55 nM T99799 C4I0CS 155533039 IC50 > 50000 nM T99799 CW1X5G 155533337 IC50 = 39000 nM T99799 C2ZAO9 155533687 IC50 = 1737.8 nM T99799 C8Q0OL 155533954 IC50 = 1100 nM T99799 CYN5O8 155534304 IC50 = 740 nM T99799 C9W7XG 155534725 IC50 = 9000 nM T99799 C76NZI 155535091 IC50 = 18000 nM T99799 CLOD29 155535170 IC50 = 500 nM T99799 CMY84N 155535601 IC50 = 27 nM T99799 CS5A6Y 155535996 IC50 = 190 nM T99799 CT90DI 155536211 IC50 = 290 nM T99799 CKI2M0 155536368 IC50 = 398.11 nM T99799 CY4D3B 155537306 IC50 = 520 nM T99799 C6R7XI 155537540 IC50 = 2.92 nM T99799 CB8CJ4 155538052 IC50 = 63 nM T99799 CA6EU8 155538194 IC50 = 15800 nM T99799 CGI1P4 155539252 IC50 = 48.6 nM T99799 C5WI2G 155539893 IC50 > 10000 nM T99799 C9JWY1 155540039 IC50 = 9360 nM T99799 C4RY7K 155540049 IC50 = 55.7 nM T99799 CRW71X 155540051 IC50 = 169 nM T99799 CM3G5X 155540209 IC50 = 7762.47 nM T99799 CVKX83 155540924 IC50 > 10000 nM T99799 CE1UC4 155541278 IC50 > 10000 nM T99799 CMT9Q2 155541386 IC50 = 70.2 nM T99799 CI64ZO 155541480 IC50 > 30000 nM T99799 CJA34X 155541507 IC50 = 48.6 nM T99799 C2PA7S 155542132 IC50 = 9.9 nM T99799 C8CM4P 155542748 IC50 = 120 nM T99799 C9KR0B 155542856 IC50 = 5310 nM T99799 CMO67L 155543176 IC50 = 568 nM T99799 CSKI49 155543595 IC50 = 86.1 nM T99799 C0RFH7 155543896 IC50 = 11.48 nM T99799 C17JEA 155543947 IC50 = 300 nM T99799 CH7ZX3 155544057 IC50 = 92.6 nM T99799 CV4MO2 155544490 IC50 = 4600 nM T99799 CNQ0F4 155544914 IC50 = 6070 nM T99799 C3FTK8 155545055 IC50 > 50000 nM T99799 CMXY60 155545085 IC50 > 10000 nM T99799 C7NA0J 155545226 IC50 = 135000 nM T99799 C79JFO 155545405 IC50 = 4520 nM T99799 C6C7AM 155545895 IC50 = 123.03 nM T99799 COW1Z3 155546180 IC50 = 6.06 nM T99799 CM6QN1 155546316 IC50 = 390 nM T99799 C35VQY 155546517 IC50 = 4520 nM T99799 C9WA1M 155546797 IC50 > 50000 nM T99799 CBPS95 155546845 IC50 > 10000 nM T99799 CPYV79 155547224 IC50 > 50000 nM T99799 CD9I8N 155547289 IC50 = 55.9 nM T99799 CX32QR 155547425 IC50 = 6.5 nM T99799 CS60BV 155547778 IC50 = 74.8 nM T99799 C4TQ5J 155548079 IC50 = 21.1 nM T99799 C5VMU7 155548207 IC50 = 21.8 nM T99799 CD8JZ5 155548223 IC50 > 30000 nM T99799 C4Q7RL 155548245 IC50 = 41.5 nM T99799 CK8RB0 155548367 IC50 = 5890000 nM T99799 C91ODF 155548523 IC50 = 910 nM T99799 CP85KA 155548858 IC50 = 480 nM T99799 CDEL58 155549426 IC50 = 26.7 nM T99799 CFT71V 155549427 IC50 = 199 nM T99799 CA8FQ3 155549571 IC50 = 1090 nM T99799 C5UC0N 155549656 IC50 = 29000 nM T99799 C94KDL 155550161 IC50 = 3.9 nM T99799 C0A7KH 155550386 IC50 = 8690 nM T99799 C2DYJ7 155551094 IC50 = 17.5 nM T99799 CAY6R5 155551298 IC50 = 27000 nM T99799 CUCF03 155551499 IC50 = 140 nM T99799 C31YDU 155551611 IC50 > 50000 nM T99799 CM2X5O 155551629 IC50 = 110 nM T99799 C5U0SM 155552824 IC50 = 93.7 nM T99799 CJXS06 155552844 IC50 = 251.19 nM T99799 CD87VC 155553046 IC50 = 0.497 nM T99799 CQ2SG6 155554219 IC50 = 6900 nM T99799 CRZW49 155554295 IC50 > 50000 nM T99799 C0P6IW 155554556 IC50 = 196 nM T99799 CS54UQ 155554734 IC50 = 1910 nM T99799 C0W3LZ 155554767 IC50 = 120 nM T99799 CFNH83 155554841 IC50 = 304 nM T99799 C8Z0MS 155555442 IC50 > 50000 nM T99799 CFK23R 155555484 IC50 = 83.7 nM T99799 C7N1YW 155555576 IC50 = 68.2 nM T99799 C53TJU 155555938 IC50 = 1148.15 nM T99799 CCHJ45 155555939 IC50 = 80.6 nM T99799 CHC64Z 155556086 IC50 = 219000 nM T99799 CD21TM 155556234 IC50 > 50000 nM T99799 C9YCT8 155556531 IC50 = 0.515 nM T99799 CD5L2W 155556671 IC50 = 9450 nM T99799 C0WAR6 155556705 IC50 = 52 nM T99799 C2EA7Q 155556733 IC50 = 1800 nM T99799 C7S5JN 155556840 IC50 = 19000 nM T99799 CDN6B5 155556926 IC50 = 9.1 nM T99799 C7IRE9 155557054 IC50 = 722 nM T99799 CU1G2L 155557132 IC50 = 1258.93 nM T99799 CK5Q9E 155557224 IC50 = 23 nM T99799 CI41HC 155557480 IC50 = 79.43 nM T99799 CVH23J 155557537 IC50 = 200 nM T99799 CVF40Y 155557821 IC50 = 25 nM T99799 CS28NH 155557943 IC50 = 13 nM T99799 CAMC16 155558019 IC50 = 50.12 nM T99799 CYP20F 155558662 IC50 > 50000 nM T99799 CE8PZ1 155559190 IC50 = 11000 nM T99799 C82GCI 155559240 IC50 = 74 nM T99799 C4T7HU 155560397 IC50 = 232 nM T99799 C0SQ7I 155560420 IC50 = 5800 nM T99799 CI8UF7 155560617 IC50 > 30000 nM T99799 C2VCE7 155560793 IC50 = 8250 nM T99799 CLY7Q6 155560920 IC50 > 30000 nM T99799 CHSY32 155560934 IC50 = 19.8 nM T99799 C95CBX 155561050 IC50 = 3900 nM T99799 CP7I9L 155561118 IC50 > 30000 nM T99799 C15FIN 155561744 IC50 = 630.96 nM T99799 CR12EX 155561772 IC50 = 4710 nM T99799 C0A9HJ 155562003 IC50 = 185 nM T99799 CCUM34 155562078 IC50 > 50000 nM T99799 CUZ64A 155562266 IC50 = 130 nM T99799 C7USO2 155562419 IC50 = 4520 nM T99799 C92PGF 155563169 IC50 = 3540 nM T99799 CJQ59S 155563181 IC50 = 7830 nM T99799 CU6NW2 155563256 IC50 = 22.9 nM T99799 CAP30C 155563421 IC50 = 4650 nM T99799 CTK04N 155563892 IC50 > 10000 nM T99799 C5HT8V 155564601 IC50 > 100000 nM T99799 CY6OR7 155564797 IC50 = 800 nM T99799 C27WPT 155565176 IC50 = 748 nM T99799 C5OTD7 155566135 IC50 = 34.67 nM T99799 C7NJY2 155566392 IC50 = 3500 nM T99799 C2NB9W 155566555 IC50 = 14000 nM T99799 CWPL14 155566983 IC50 = 68000 nM T99799 C9R2MS 155567099 IC50 = 78 nM T99799 CNQ18H 155567205 IC50 = 6.95 nM T99799 CM63EC 155567324 IC50 = 39.81 nM T99799 C40XPW 155567716 IC50 = 29000 nM T99799 CW3Q7C 155567905 IC50 = 22 nM T99799 C3EPS6 155567920 IC50 = 35.6 nM T99799 CG3BR0 155567943 IC50 > 100000 nM T99799 CRMO93 155567970 IC50 = 7.8 nM T99799 CR24FZ 155568280 IC50 = 600 nM T99799 CJLF85 155568310 IC50 > 50000 nM T99799 CF1J8X 155568638 IC50 > 50000 nM T99799 CDQ05E 155568688 IC50 = 20 nM T99799 C10CZA 155569041 IC50 = 75.7 nM T99799 CZGB74 155569334 IC50 = 65.7 nM T99799 C1YG5A 10015862 IC50 = 138 nM T99799 CB49KJ 10906319 IC50 = 23780 nM T99799 D00AHD 44435223 Ki = 3.5 nM T99799 D00ANJ 1897797 Ki > 100000 nM T99799 D00DKI 10107976 IC50 = 153 nM T99799 D00KTT 44568318 Ki = 18100 nM T99799 D00MFR 44419695 IC50 = 1099.01 nM T99799 D00PLH 44428832 Ki > 100000 nM T99799 D00QLR 10403152 IC50 = 1370 nM T99799 D00RIX 5280443 Ki = 37400 nM T99799 D00VXE 3253193 Ki = 350 nM T99799 D00XHC 12851057 Ki = 180 nM T99799 D01AJQ 46232725 IC50 = 400 nM T99799 D01EZC 44421938 IC50 = 2650 nM T99799 D01FNH 24905597 Ki = 2260 nM T99799 D01HRG 12884 Ki = 68800 nM T99799 D01HZN 44428835 Ki > 100000 nM T99799 D01LVY 3473393 Ki = 2500 nM T99799 D01MAC 25133941 IC50 = 894 nM T99799 D01OND 46080 IC50 = 18000 nM T99799 D01QRR 25130201 IC50 = 6 nM T99799 D01VAU 123493 Ki > 100000 nM T99799 D01VCS 44428837 Ki > 100000 nM T99799 D01XGP 123358 Ki = 2630 nM T99799 D01XKY 3473392 Ki = 1300 nM T99799 D02BDL 8433 Ki > 100000 nM T99799 D02DUJ 65719 IC50 = 12 nM T99799 D02GJG 11043027 Ki > 100000 nM T99799 D02HQS 19377173 Ki > 100000 nM T99799 D02LWX 44419700 IC50 = 8700 nM T99799 D02SGJ 19009 IC50 > 100000 nM T99799 D02TLP 11363 Ki > 100000 nM T99799 D02XHM 44421959 IC50 = 100 nM T99799 D02YSX 197033 IC50 = 7900000 nM T99799 D03HZT 89076 Ki > 100000 nM T99799 D03NTO 25129142 IC50 = 57 nM T99799 D03OGO 465614 IC50 = 770 nM T99799 D03TPH 87203 Ki > 100000 nM T99799 D04AWS 704267 Ki = 2990 nM T99799 D04AXR 96047 Ki > 100000 nM T99799 D04CDV 44428829 Ki > 100000 nM T99799 D04CTO 44435201 Ki = 1700 nM T99799 D04EXR 251908 Ki > 100000 nM T99799 D04FHZ 9906452 IC50 = 1950 nM T99799 D04GTP 23645738 IC50 = 1700 nM T99799 D04IXN 16645663 Ki = 10500 nM T99799 D04JCW 25128787 IC50 = 700 nM T99799 D04PKD 25129847 IC50 = 980 nM T99799 D04SYM 25129843 IC50 = 5100 nM T99799 D04ZWS 11173982 IC50 = 260 nM T99799 D04ZZU 24905653 Ki = 570 nM T99799 D05AVX 60983 Ki > 100000 nM T99799 D05DIN 24905595 Ki = 340 nM T99799 D05EMT 22574258 Ki > 100000 nM T99799 D05EYA 18946 Ki > 100000 nM T99799 D05GPI 44421960 IC50 = 120 nM T99799 D05LTW 22574224 Ki = 1270 nM T99799 D05PNO 4135273 Ki > 100000 nM T99799 D05QFR 25133942 IC50 = 2500 nM T99799 D05UJV 52945624 IC50 = 16000 nM T99799 D05VLV 3473842 Ki = 1900 nM T99799 D05VUC 19971657 Ki > 100000 nM T99799 D05XPW 46232686 IC50 = 1220 nM T99799 D05XRY 2752926 Ki > 100000 nM T99799 D05ZCX 44435802 Ki > 100000 nM T99799 D06BDB 25128786 IC50 = 4100 nM T99799 D06ERH 637760 IC50 = 87000 nM T99799 D06FFD 96430 Ki > 100000 nM T99799 D06GYH 16745302 Ki > 100000 nM T99799 D06KQH 10178151 IC50 = 1580 nM T99799 D06UXW 107759 IC50 = 977.24 nM T99799 D06VGD 6724 Ki = 2970 nM T99799 D06YEB 44435197 Ki = 1700 nM T99799 D06ZRX 5281717 IC50 = 2950 nM T99799 D07AYF 3107576 Ki = 10200 nM T99799 D07CFJ 589576 Ki > 100000 nM T99799 D07EDG 1901244 Ki = 12600 nM T99799 D07RIQ 71028 IC50 > 10000 nM T99799 D07YJG 11351920 IC50 = 7000 nM T99799 D08AOG 90571 Ki > 100000 nM T99799 D08BKE 44568822 IC50 = 359 nM T99799 D08FQW 24905593 Ki = 1690 nM T99799 D08NNF 46229054 Ki = 10000 nM T99799 D08PWL 52945680 IC50 = 70000 nM T99799 D08TBI 24905535 Ki = 3190 nM T99799 D08UET 4939 IC50 = 13200 nM T99799 D08UOB 44428840 Ki > 100000 nM T99799 D08XQI 9395 IC50 = 7 nM T99799 D08ZLS 705757 Ki = 4450 nM T99799 D09ALJ 5280805 Ki = 501200 nM T99799 D09CGV 44419702 IC50 = 1625.55 nM T99799 D09DWA 3473839 Ki = 3100 nM T99799 D09GKY 705769 Ki = 2810 nM T99799 D09GXM 44421953 IC50 = 800 nM T99799 D09HZE 705776 Ki = 7100 nM T99799 D09LSR 11437501 Ki > 100000 nM T99799 D09OPL 705775 Ki = 1560 nM T99799 D09QDC 5420 IC50 = 733 nM T99799 D09YLY 25129143 IC50 = 88 nM T99799 D0A0YX 5143 IC50 = 3600 nM T99799 D0A5FO 222149 Ki = 220 nM T99799 D0AQ3K 44421955 IC50 = 100 nM T99799 D0AW4P 10868634 Ki > 100000 nM T99799 D0B0ZM 2235291 Ki = 430 nM T99799 D0B1TQ 1810509 Ki > 100000 nM T99799 D0B4DT 44421954 IC50 = 80 nM T99799 D0B6IQ 2301676 Ki = 9200 nM T99799 D0B8YX 75511 Ki > 100000 nM T99799 D0BB2U 2385968 Ki > 100000 nM T99799 D0C0XU 10496398 IC50 = 40 nM T99799 D0C1LI 53378764 IC50 = 1820 nM T99799 D0C9AD 277990 Ki = 21900 nM T99799 D0CN8Z 11392969 Ki > 100000 nM T99799 D0D0BI 8371 Ki = 268 nM T99799 D0D2HH 44428834 Ki > 100000 nM T99799 D0D7FN 283893 Ki > 100000 nM T99799 D0D7MN 44435217 Ki = 88 nM T99799 D0D8IH 777336 Ki = 310 nM T99799 D0DB9T 704261 Ki = 10600 nM T99799 D0DR7A 934131 Ki = 12100 nM T99799 D0DV9Z 44419694 IC50 = 20900 nM T99799 D0DW9J 123072 Ki > 100000 nM T99799 D0E2IG 44428839 Ki > 100000 nM T99799 D0E4GM 16728608 IC50 = 3600 nM T99799 D0E5ZP 604575 Ki > 100000 nM T99799 D0EI5V 16115140 IC50 = 40000 nM T99799 D0EK7H 2734793 Ki > 100000 nM T99799 D0EQ1Z 45487256 IC50 = 1.2 nM T99799 D0ER5C 44419701 IC50 = 32200 nM T99799 D0F3QP 5889042 IC50 = 2570 nM T99799 D0F3RN 89801 Ki > 100000 nM T99799 D0F5EJ 11375002 IC50 = 10.8 nM T99799 D0F5VY 94860 Ki = 1670 nM T99799 D0FO2B 1923 IC50 > 100 nM T99799 D0FP5F 46232685 IC50 = 10400 nM T99799 D0G0ED 44420671 IC50 = 790 nM T99799 D0G0GZ 19916609 Ki = 18300 nM T99799 D0G2DQ 4669250 Ki > 100000 nM T99799 D0G2WI 10318177 IC50 = 4500 nM T99799 D0G3TK 5280863 Ki = 43100 nM T99799 D0G5TL 44419706 IC50 = 2685.34 nM T99799 D0H1NU 10135721 IC50 = 3520 nM T99799 D0H2UG 52946279 IC50 = 360 nM T99799 D0H3BC 44421943 IC50 = 2490 nM T99799 D0H3WJ 44435193 Ki = 560 nM T99799 D0I3XA 6422124 IC50 = 77300 nM T99799 D0I4LX 1403 IC50 = 3370 nM T99799 D0I5LV 24905596 Ki = 710 nM T99799 D0I7BX 16645664 Ki = 36 nM T99799 D0IC5U 11573367 IC50 = 3.6 nM T99799 D0J1IX 1238015 Ki = 610 nM T99799 D0J3SN 1868 IC50 > 10000 nM T99799 D0J5AU 25133940 IC50 = 3900 nM T99799 D0J8LQ 607810 Ki = 600 nM T99799 D0JH7C 72810 Ki > 100000 nM T99799 D0JI0H 3542734 Ki = 28100 nM T99799 D0K3YM 704259 Ki = 3410 nM T99799 D0K6OM 44428838 Ki > 100000 nM T99799 D0K6PO 316765 Ki > 100000 nM T99799 D0K7EC 705771 Ki = 1050 nM T99799 D0K8BT 25129490 IC50 = 669 nM T99799 D0L1EI 9969234 IC50 = 1890 nM T99799 D0L1ST 2777298 Ki > 100000 nM T99799 D0L3EE 262319 Ki = 5800 nM T99799 D0L4MF 44428833 Ki > 100000 nM T99799 D0L4OW 9823294 IC50 = 310 nM T99799 D0L5QJ 11408144 IC50 = 6000 nM T99799 D0L9YJ 44421937 IC50 = 8330 nM T99799 D0LJ2F 11806279 Ki > 100000 nM T99799 D0LL8H 25129141 IC50 = 4.3 nM T99799 D0M0BM 10399068 IC50 = 114 nM T99799 D0M2EM 4650 Ki = 2050 nM T99799 D0M2LD 1476756 IC50 > 1000000 nM T99799 D0M2TY 10168 IC50 = 17000 nM T99799 D0M2ZD 44428831 Ki > 100000 nM T99799 D0M4IE 9549196 Ki = 0.163 nM T99799 D0M5NR 3794313 Ki > 100000 nM T99799 D0M6IJ 44435218 Ki = 470 nM T99799 D0MF5Y 5281614 Ki = 90000 nM T99799 D0N0HK 73252 Ki = 3200 nM T99799 D0N6XS 44435196 Ki = 400 nM T99799 D0N8YZ 2427416 Ki > 100000 nM T99799 D0N9ZR 1718647 Ki = 56500 nM T99799 D0NJ4G 80771 Ki > 100000 nM T99799 D0NJ5W 10055202 IC50 = 11600 nM T99799 D0O0LU 264734 Ki > 100000 nM T99799 D0O2OH 9907847 IC50 = 50 nM T99799 D0O8DZ 44421948 IC50 = 1430 nM T99799 D0O8LK 16066832 IC50 = 150 nM T99799 D0O9YQ 52941983 IC50 = 1000 nM T99799 D0OJ9P 49799304 IC50 = 550 nM T99799 D0P1IK 44428841 Ki > 100000 nM T99799 D0P3VH 893336 Ki = 6200 nM T99799 D0P7TN 465615 IC50 = 4600 nM T99799 D0PF7F 9928397 IC50 = 1950 nM T99799 D0PQ5R 24905594 Ki = 2850 nM T99799 D0Q0BV 24905710 Ki = 120 nM T99799 D0Q2YJ 6763 Ki = 190 nM T99799 D0Q3EV 52948017 IC50 = 120 nM T99799 D0R2GR 46229025 Ki = 2660 nM T99799 D0R2QC 10275242 IC50 = 31550 nM T99799 D0S1MC 23643351 IC50 = 118000 nM T99799 D0S2DW 9844749 IC50 = 48900 nM T99799 D0S3WF 10222714 IC50 = 1350 nM T99799 D0S6TW 1845 Ki > 100000 nM T99799 D0S8AS 44568319 Ki = 4300 nM T99799 D0S9YA 638276 IC50 = 84000 nM T99799 D0SP2O 7054 Ki > 100000 nM T99799 D0T3PW 5281672 Ki = 71000 nM T99799 D0T5MD 25128788 IC50 = 334 nM T99799 D0T5XC 31494 Ki > 100000 nM T99799 D0U0BV 44428830 Ki > 100000 nM T99799 D0U3JD 16358 Ki > 100000 nM T99799 D0U7BQ 24905592 Ki = 390 nM T99799 D0U9AU 11385845 IC50 = 6 nM T99799 D0UK5A 76996 Ki > 100000 nM T99799 D0UT1X 101375 Ki > 100000 nM T99799 D0UZ8R 71043 Ki > 100000 nM T99799 D0V4RD 3112604 Ki = 820 nM T99799 D0V7EK 3773589 Ki = 570 nM T99799 D0V8PE 24905534 Ki = 13400 nM T99799 D0W4WB 25129492 IC50 = 3700 nM T99799 D0W9VA 10667 Ki = 2290 nM T99799 D0WB1D 10221700 IC50 = 560 nM T99799 D0WH4J 25129844 IC50 = 639 nM T99799 D0WX6R 3477013 Ki = 3100 nM T99799 D0X0ER 344135 Ki = 30600 nM T99799 D0X4HG 10765787 IC50 = 48 nM T99799 D0X7CW 497286 IC50 = 350 nM T99799 D0XI4U 5319470 IC50 = 17458.22 nM T99799 D0XL1R 9976105 IC50 = 2915 nM T99799 D0Y0UV 19916610 Ki = 710 nM T99799 D0Y0XQ 2779383 Ki > 100000 nM T99799 D0Y2TE 10112356 IC50 = 5230 nM T99799 D0Y5KN 44568823 IC50 = 72 nM T99799 D0Y6RZ 22574214 Ki > 100000 nM T99799 D0Y7FX 8651 Ki > 100000 nM T99799 D0Y7HG 5281616 Ki = 6900 nM T99799 D0YZ3E 44435200 Ki = 220 nM T99799 D0Z1WQ 76915 Ki > 100000 nM T99799 D0Z5KQ 8400 Ki > 100000 nM T99799 D0Z6CZ 5139980 Ki > 100000 nM T99799 D0Z6DK 44423026 IC50 > 50000 nM T99799 D0Z6WU 201563 IC50 = 5000 nM T99799 D0Z8HX 16786802 Ki > 100000 nM T99799 D0ZI7F 211174 IC50 = 17400 nM T99799 D0ZL6B 3772674 Ki > 100000 nM T99799 D0ZR2T 2732752 Ki > 100000 nM T99799 D0ZT5C 44428828 Ki > 100000 nM T11911 CV4Q5S 704452 IC50 = 4 nM T11911 CDK30S 772885 IC50 = 43 nM T11911 CD8AV5 9852584 IC50 = 3 nM T11911 CA8L5J 10372090 IC50 = 1 nM T11911 C67LUP 24857841 IC50 = 3800 nM T11911 C6CZ1L 25110719 IC50 = 300 nM T11911 CJ2AK1 44589880 IC50 = 1190 nM T26428 CIG85H 11282247 IC50 > 10000 nM T26428 CQF60E 11386451 IC50 = 171 nM T26428 CBJ68T 11396908 IC50 = 626 nM T26428 CJI4A8 11397595 IC50 = 516 nM T26428 CF6XZ1 11419337 IC50 = 104 nM T26428 C98ADL 11454184 IC50 = 178 nM T26428 CKU5J7 11464405 IC50 = 25 nM T26428 CMQ86R 11495432 IC50 = 66 nM T26428 CCP2Z0 11510399 IC50 = 57 nM T26428 CD4PM0 11518159 IC50 = 7140 nM T26428 COT53B 11518384 IC50 = 1120 nM T26428 CZD24Q 11554412 IC50 = 44 nM T26428 CZ6C8H 11583193 IC50 = 46 nM T26428 COE14C 11589812 IC50 = 110 nM T26428 CS28HA 11612403 IC50 = 654 nM T26428 CJQK24 11647458 IC50 = 106 nM T26428 C1F9VA 11662657 IC50 = 26 nM T26428 CIZQ65 11711452 IC50 = 35 nM T26428 C74DRE 11719291 IC50 = 162 nM T26428 CDT5W6 11775399 IC50 = 11 nM T26428 CJ51DI 11973802 IC50 > 10000 nM T26428 C7K5AW 16721015 IC50 = 15 nM T26428 CS2H5L 44402329 IC50 = 275 nM T26428 C45JVO 44402350 IC50 = 2880 nM T26428 C8OVR3 44402414 IC50 > 10000 nM T26428 CVA21D 44402419 IC50 > 10000 nM T26428 C5FDU2 44402420 IC50 > 10000 nM T26428 C1HVF7 44402433 IC50 > 10000 nM T26428 CF2XD9 44402484 IC50 > 10000 nM T26428 CQN5D8 44402505 IC50 = 1177 nM T26428 CBEX17 44402535 IC50 > 10000 nM T26428 CH4R7K 44402549 IC50 > 10000 nM T26428 C04HCO 44402563 IC50 = 751 nM T26428 CKE6L3 44402567 IC50 = 894 nM T26428 CA3L4O 44402593 IC50 > 10000 nM T26428 CDRU68 44402599 IC50 > 10000 nM T26428 CVZB43 44402635 IC50 > 10000 nM T26428 C8K1GV 44402677 IC50 = 147 nM T26428 C0NWZ9 44402768 IC50 = 1810 nM T26428 CPE50S 44417890 IC50 = 2750 nM T26428 CL5XO4 44417897 IC50 = 173 nM T26428 CM9QI8 44417899 IC50 = 95 nM T26428 CI16UJ 44417902 IC50 > 10000 nM T26428 C9BDI1 44417906 IC50 = 1380 nM T26428 CN2G7U 44417910 IC50 = 569 nM T26428 CH08OA 44417936 IC50 = 5590 nM T26428 C7W8KZ 44417937 IC50 = 2410 nM T26428 CH3QM1 44417938 IC50 = 551 nM T26428 CP1U0Z 44417939 IC50 = 233 nM T26428 D05UZY 11539096 IC50 = 29 nM T20371 D09VBC 2562 IC50 = 32 nM T20371 D01RBE 54670732 IC50 = 0.5 nM T20371 D03GPW 54577783 IC50 = 0.44 nM T20371 D05NQZ 57404019 IC50 = 3.2 nM T20371 D0AF0O 54670056 IC50 = 0.079 nM T20371 D0LZ4A 57393568 IC50 = 0.49 nM T20371 D01KIU 126402 IC50 = 100000 nM T20371 D01XGX 178060 IC50 > 100000 nM T20371 D02KLW 180081 IC50 = 5.3 nM T20371 C5NKT4 15362 IC50 > 30000 nM T20371 CER1X5 50471 IC50 = 4400 nM T20371 CO08EI 98468 IC50 = 1000 nM T20371 COT8I4 100137 IC50 = 1900 nM T20371 C2DQG8 114745 Ki = 16 nM T20371 CSL8T0 129016 IC50 > 30000 nM T20371 CU2RH4 202478 IC50 = 100000 nM T20371 CWXD84 231173 IC50 = 3800 nM T20371 CHT75C 251645 IC50 = 24000 nM T20371 C6BQD9 411452 IC50 > 30000 nM T20371 CJ9FW1 583452 IC50 = 11000 nM T20371 CEK87Y 583453 IC50 = 12000 nM T20371 C9Q3AH 611407 IC50 = 4270 nM T20371 C07PSU 4236593 IC50 > 30000 nM T20371 C3O1DG 10354345 IC50 = 117500 nM T20371 C2YP3V 10727124 IC50 = 3900 nM T20371 CST50C 11770665 IC50 = 5300 nM T20371 CJNM07 13049800 IC50 = 20000 nM T20371 C92OAS 14494163 IC50 > 30000 nM T20371 C9H3EI 14548157 IC50 = 2300 nM T20371 C6ZQH1 14548158 IC50 = 4900 nM T20371 C2E1WD 14548159 IC50 = 9500 nM T20371 C35XWF 14548160 IC50 > 30000 nM T20371 C41PLQ 14548162 IC50 = 6200 nM T20371 CPL8H6 14548163 IC50 > 30000 nM T20371 CAO15G 14548166 IC50 = 5400 nM T20371 CQYL12 44274582 IC50 = 760 nM T20371 C0AHE3 44362525 IC50 = 107000 nM T20371 C74MNU 49781061 IC50 = 4090 nM T20371 CKT80S 49781062 IC50 = 352 nM T20371 C13BKE 49781063 IC50 = 56 nM T20371 CX6V0Z 49781064 IC50 = 122 nM T20371 C7H5GL 49781278 IC50 = 49 nM T20371 CTE79O 49781279 IC50 = 72 nM T20371 C4J0TS 49781280 IC50 = 73 nM T20371 C5PM9X 49781281 IC50 = 300 nM T20371 C4H8OK 49782407 IC50 = 158 nM T20371 CT1C4W 49782408 IC50 = 79 nM T20371 CUO8P9 49782614 IC50 = 308 nM T20371 C9HDP1 49782615 IC50 = 24 nM T20371 CC1PQ4 49782616 IC50 = 4 nM T20371 CB6F0L 49782617 IC50 = 54 nM T20371 CMR0U7 49782849 IC50 = 9 nM T20371 CDH5C3 49782850 IC50 = 21 nM T20371 C2OH5D 49782851 IC50 = 3 nM T20371 CH97YZ 49782852 IC50 = 5 nM T20371 CK5UZ9 49782853 IC50 = 2 nM T20371 CU14ZN 49783051 IC50 = 4 nM T20371 C50SVG 49783052 IC50 = 1 nM T20371 CD9E8U 49783053 IC50 = 37 nM T20371 C1WGZ4 49783054 IC50 = 10 nM T20371 COX12Q 49783055 IC50 = 2 nM T20371 CNPM04 49783265 IC50 = 21 nM T20371 CDN20Q 49783266 IC50 = 5 nM T20371 CR86KI 49783267 IC50 = 12 nM T20371 C07TLJ 51003394 IC50 = 3.7 nM T20371 CBRG85 51003395 IC50 = 2.3 nM T20371 CV6CR5 51003396 IC50 = 4.7 nM T20371 CMZ50Q 51003397 IC50 = 7 nM T20371 CWR84J 51003599 IC50 = 1.1 nM T20371 C7OY8A 51003600 IC50 = 12 nM T20371 CAMJ95 51003601 IC50 = 1.7 nM T20371 C09ACM 52941183 IC50 = 432 nM T20371 CIS3X9 52941184 IC50 = 300 nM T20371 CZ5GN7 52941192 IC50 = 4370 nM T20371 CMXQ50 52941193 IC50 = 32000 nM T20371 C3I6HF 52941487 IC50 = 800 nM T20371 CHE98D 52942383 IC50 = 27000 nM T20371 CP3T7C 52942396 IC50 = 68 nM T20371 CJ0N5T 52942838 IC50 = 23000 nM T20371 C79QCT 52942912 IC50 = 570 nM T20371 CD6SG7 52943599 IC50 = 518 nM T20371 CK8AG6 52944766 IC50 = 280000 nM T20371 C8V4CB 52944768 IC50 = 78000 nM T20371 CN29BT 52944799 IC50 = 21000 nM T20371 C8EV4H 52945123 IC50 = 240 nM T20371 C7S0LM 52945988 IC50 = 184000 nM T20371 CQG9D2 52945989 IC50 = 146000 nM T20371 CVE41W 52946012 IC50 = 22 nM T20371 C3Y5ML 52946014 IC50 = 1200 nM T20371 C0D4YX 52946016 IC50 = 338000 nM T20371 C4PL8G 52946024 IC50 = 320000 nM T20371 CDIB63 52946037 IC50 = 399 nM T20371 C2AEP8 52947234 IC50 = 221000 nM T20371 C72WZK 52947236 IC50 = 163000 nM T20371 CA7MX6 52947259 IC50 = 5000 nM T20371 CKZ3I8 52947260 IC50 = 710000 nM T20371 CR0NY1 52947569 IC50 = 90 nM T20371 C25PHE 52947570 IC50 = 849 nM T20371 CO3T2A 52948472 IC50 = 476000 nM T20371 C4I5ZC 52948473 IC50 = 92000 nM T20371 C8FWU2 52948785 IC50 = 850 nM T20371 C2QUJ4 52948786 IC50 = 6200 nM T20371 C1E4WF 52949672 IC50 = 223 nM T20371 CAJ4K3 52949696 IC50 = 827000 nM T20371 CJ1HS0 52949698 IC50 = 74000 nM T20371 CFZN43 52949699 IC50 = 274000 nM T20371 CO27HZ 53317386 IC50 = 22 nM T20371 CT6I2E 53317387 IC50 = 17 nM T20371 CT03AI 53317388 IC50 = 32 nM T20371 CF7TW1 53318672 IC50 = 155 nM T20371 CCF6W3 53318673 IC50 = 25 nM T20371 CECL97 53319995 IC50 = 25 nM T20371 CA2HR7 53319997 IC50 = 129 nM T20371 CAQ1Y6 53319998 IC50 = 18 nM T20371 C5X1PK 53321296 IC50 = 18 nM T20371 CV0D5S 53321297 IC50 = 34 nM T20371 CE3H8K 53322625 IC50 = 42 nM T20371 CW1Q7R 53324275 IC50 = 30 nM T20371 C0JSE4 53325246 IC50 = 10 nM T20371 C1CD3T 53325247 IC50 = 71 nM T20371 CN9CQ6 53325248 IC50 = 21 nM T20371 CTU2Q0 53325249 IC50 = 93 nM T20371 C9XWN6 53325250 IC50 = 44 nM T20371 C8YP0W 53325251 IC50 = 13 nM T20371 CC7R9A 53325252 IC50 = 19 nM T20371 C2M9NY 53326527 IC50 = 141 nM T20371 C7YM6N 53326528 IC50 = 16 nM T20371 CO9V2U 53326529 IC50 = 64 nM T20371 CY7R8D 53326530 IC50 = 24 nM T20371 CX0JV4 53326531 IC50 = 8.5 nM T20371 C7TLQ6 53326532 IC50 = 15 nM T20371 C7V1HI 53326533 IC50 = 27 nM T20371 C9PB3D 54577781 IC50 = 0.78 nM T20371 CGF49X 54577784 IC50 = 1.2 nM T20371 C57DQW 54670057 IC50 = 0.66 nM T20371 C7L5YB 54670058 IC50 = 2.6 nM T20371 CM7FC6 54670152 IC50 = 16.7 nM T20371 CS6V7K 54769300 IC50 = 11 nM T20371 C9V1KU 54769301 IC50 = 6.4 nM T20371 CLAF98 54769527 IC50 = 18 nM T20371 CG7L0F 54769529 IC50 = 0.2 nM T20371 C0BY9H 54769530 IC50 = 2.8 nM T20371 CUI25K 54769531 IC50 = 0.3 nM T20371 CME93J 56835036 IC50 = 1.5 nM T20371 C0X4GE 57334109 IC50 = 0.37 nM T20371 CQ67NY 57336186 IC50 = 350 nM T20371 C85GTH 57390647 IC50 = 15 nM T20371 C1DB0V 57390648 IC50 = 17 nM T20371 C7JP8I 57390709 IC50 = 151 nM T20371 CS48ZL 57390759 IC50 = 509 nM T20371 CX83BE 57390760 IC50 = 190 nM T20371 C78RGH 57390761 IC50 = 333 nM T20371 CWQX89 57390800 IC50 = 2553 nM T20371 C3KP1N 57390801 IC50 = 3449 nM T20371 CCM7G0 57390885 IC50 = 998 nM T20371 CM14QA 57390886 IC50 > 10000 nM T20371 CPR98A 57390952 IC50 = 10 nM T20371 CL93GA 57390953 IC50 = 5 nM T20371 CAPZ29 57390954 IC50 = 181 nM T20371 CM8D3F 57392437 IC50 = 37 nM T20371 CFG42K 57392438 IC50 = 11 nM T20371 CYJI47 57392439 IC50 = 53 nM T20371 C8RCG0 57392440 IC50 = 80 nM T20371 CP5MU3 57392441 IC50 = 1.4 nM T20371 C4IL5F 57392442 IC50 = 79 nM T20371 C95CVX 57392511 IC50 = 17 nM T20371 CQK9X5 57392570 IC50 = 537 nM T20371 C9ZG8C 57392571 IC50 = 32 nM T20371 C8DN3X 57392616 IC50 = 828 nM T20371 CVDQ72 57392617 IC50 = 3623 nM T20371 CYCK96 57392697 IC50 = 48 nM T20371 C23OQN 57392698 IC50 > 10000 nM T20371 CT3W6N 57393567 IC50 = 3.2 nM T20371 C1JD4W 57394149 IC50 = 2.7 nM T20371 C2AC1D 57394150 IC50 = 21 nM T20371 CXQ3R4 57394151 IC50 = 2.5 nM T20371 CHMX49 57394152 IC50 = 10 nM T20371 CKV8Y2 57394153 IC50 = 2.8 nM T20371 C8R7AK 57394220 IC50 = 1520 nM T20371 CI25ZB 57394292 IC50 = 28 nM T20371 CFC3D6 57394293 IC50 = 21 nM T20371 CC2L5N 57394294 IC50 = 58 nM T20371 CE63JL 57394295 IC50 = 7922 nM T20371 CVK4H6 57394296 IC50 = 15 nM T20371 C2B7FH 57394336 IC50 = 3882 nM T20371 CVU24A 57394402 IC50 > 10000 nM T20371 CP1UM3 57394403 IC50 > 10000 nM T20371 CZ0BQ1 57394469 IC50 = 427 nM T20371 C89OBN 57395279 IC50 = 15.6 nM T20371 CZH4R9 57395934 IC50 = 32 nM T20371 C2QZP8 57395935 IC50 = 1.7 nM T20371 CSGZ32 57395936 IC50 = 5.2 nM T20371 CMP0V3 57395937 IC50 = 2.1 nM T20371 CH6G8V 57396046 IC50 = 286 nM T20371 COH93L 57396047 IC50 = 5541 nM T20371 CR6J8O 57396048 IC50 = 87 nM T20371 C9SQO2 57396049 IC50 = 44 nM T20371 C4LEU7 57396166 IC50 = 0.74 nM T20371 CAN37H 57396167 IC50 = 1 nM T20371 CPAV25 57396168 IC50 = 374 nM T20371 C1D5PJ 57396228 IC50 = 5.6 nM T20371 CVN1L5 57397048 IC50 = 23 nM T20371 C2K6VP 57397049 IC50 = 4.5 nM T20371 C4OX0M 57397050 IC50 = 1.9 nM T20371 CDQS60 57397051 IC50 = 200 nM T20371 C0RDU5 57397724 IC50 = 33 nM T20371 CWTV16 57397725 IC50 = 3.8 nM T20371 CU98FN 57397726 IC50 = 8.4 nM T20371 CEV05L 57397847 IC50 = 42 nM T20371 CB7Z0W 57397848 IC50 = 130 nM T20371 CL5GE3 57397902 IC50 = 8264 nM T20371 C3J9GE 57397903 IC50 = 1524 nM T20371 CX1ED2 57397982 IC50 = 0.17 nM T20371 CZA65K 57398810 IC50 = 1.9 nM T20371 C7FGO0 57399385 IC50 = 7.6 nM T20371 CPB52Q 57399386 IC50 = 64 nM T20371 CS78WX 57399387 IC50 = 26 nM T20371 CA9N5U 57399388 IC50 = 45 nM T20371 CC2UF6 57399389 IC50 = 1250 nM T20371 CAD4J8 57399390 IC50 = 3.8 nM T20371 CZ04HU 57399391 IC50 = 0.3 nM T20371 CS0IB1 57399392 IC50 = 11 nM T20371 CCUL27 57399452 IC50 = 313 nM T20371 CK2HB3 57399507 IC50 = 91 nM T20371 CJ9R8O 57399508 IC50 = 241 nM T20371 CMC27V 57399509 IC50 = 91 nM T20371 CL95JG 57399510 IC50 = 54 nM T20371 CE2Q5M 57399511 IC50 = 1704 nM T20371 CB7LT9 57399550 IC50 = 575 nM T20371 CF1VY2 57399551 IC50 > 10000 nM T20371 CW83EX 57399625 IC50 = 102 nM T20371 CNV8K2 57399626 IC50 = 225 nM T20371 C2XHT7 57399683 IC50 = 38 nM T20371 CS09AD 57400492 IC50 = 3.4 nM T20371 CWDB98 57400493 IC50 = 9.5 nM T20371 C92PQX 57400494 IC50 = 8.3 nM T20371 CD1YE3 57401142 IC50 = 0.9 nM T20371 C4RC9H 57401143 IC50 = 0.6 nM T20371 CC1R3I 57401144 IC50 = 199 nM T20371 CM0J3V 57401145 IC50 = 3.2 nM T20371 C60LMR 57401146 IC50 = 1.2 nM T20371 CJCM54 57401212 IC50 = 21 nM T20371 C9H2KX 57401386 IC50 = 160 nM T20371 CAQI49 57401387 IC50 = 60 nM T20371 CIY78W 57401444 IC50 = 16 nM T20371 CJ09EF 57401445 IC50 = 14 nM T20371 C8R7GF 57402296 IC50 = 41 nM T20371 C2QLS0 57402297 IC50 = 474 nM T20371 C9WA0C 57402298 IC50 = 54 nM T20371 CEPX74 57402299 IC50 = 1 nM T20371 C7R1IA 57402300 IC50 = 1.6 nM T20371 CWL9K7 57402301 IC50 = 0.73 nM T20371 COWR29 57402919 IC50 = 26 nM T20371 C1M2UL 57402920 IC50 = 15 nM T20371 C1HS8N 57402960 IC50 = 8700 nM T20371 CF3I4X 57402961 IC50 = 104 nM T20371 CPF45C 57403008 IC50 = 839 nM T20371 CV7IC6 57403009 IC50 = 1024 nM T20371 C60MVW 57403010 IC50 = 52 nM T20371 CFB61E 57403059 IC50 = 2290 nM T20371 CHJ83M 57403133 IC50 = 6.6 nM T20371 CS8ND6 57403134 IC50 = 2.6 nM T20371 C4KI5Y 57403884 IC50 = 6 nM T20371 C76ZJN 57404018 IC50 = 11 nM T20371 C1W7KP 57404020 IC50 = 169 nM T20371 CN56WD 57404021 IC50 = 84 nM T20371 C8T4IB 68199725 IC50 = 12 nM T20371 C73IYJ 68199726 IC50 = 2.7 nM T20371 CV0P7D 68199727 IC50 = 36 nM T20371 CY41JC 68199728 IC50 = 4.6 nM T20371 C1NIP0 68199729 IC50 = 480 nM T20371 C80ARK 68199735 IC50 = 0.18 nM T20371 C7NM8D 68199737 IC50 = 0.6 nM T20371 CZ3LH9 68199741 IC50 = 0.95 nM T20371 C3TIW0 68199753 IC50 = 17 nM T20371 CZE0W7 70681372 IC50 = 0.2 nM T20371 C3TBU2 70681399 IC50 = 14 nM T20371 CMB09P 70681439 IC50 = 13 nM T20371 C20TWB 70681611 IC50 = 6.4 nM T20371 CJS65Q 70681624 IC50 = 12.1 nM T20371 CS2YJ9 70681625 IC50 = 2.7 nM T20371 C8TM3A 70683496 IC50 = 1.4 nM T20371 C45LNR 70683497 IC50 = 1 nM T20371 CK12GS 70683498 IC50 = 11 nM T20371 CQ5AH6 70683558 IC50 = 2.5 nM T20371 CBG28Q 70683752 IC50 = 0.4 nM T20371 C4YDR2 70683753 IC50 = 2 nM T20371 CR7V9L 70685575 IC50 = 1 nM T20371 C2AQ6E 70685576 IC50 = 6.7 nM T20371 C43VWQ 70685577 IC50 = 0.4 nM T20371 CI5O8T 70685597 IC50 = 12 nM T20371 CUPI59 70685598 IC50 = 315 nM T20371 C9XPD0 70687722 IC50 = 815 nM T20371 CRF46T 70687723 IC50 = 3070 nM T20371 CL7N9S 70687749 IC50 = 4.3 nM T20371 CD7S8H 70687815 IC50 = 5.6 nM T20371 CAC97E 70688019 IC50 = 49.9 nM T20371 CBFP89 70688020 IC50 = 6 nM T20371 CQ0WP3 70688021 IC50 = 24.7 nM T20371 C45FZR 70688022 IC50 = 0.8 nM T20371 CPW14Y 70689768 IC50 = 10 nM T20371 CW1N2K 70689769 IC50 = 0.7 nM T20371 C54NPT 70689770 IC50 = 100 nM T20371 CZFE74 70689771 IC50 = 852 nM T20371 CREJ45 70689799 IC50 = 33 nM T20371 CMZC24 70690050 IC50 = 1.6 nM T20371 CJKT71 70690051 IC50 = 2 nM T20371 C63LPU 70690052 IC50 = 44.3 nM T20371 C52BLV 70690053 IC50 = 28 nM T20371 C08KGO 70690054 IC50 = 0.9 nM T20371 C0OCY6 70690055 IC50 = 635 nM T20371 C20PBJ 70691913 IC50 = 1 nM T20371 CFY27L 70691914 IC50 = 10 nM T20371 CU7HW9 70691939 IC50 = 0.5 nM T20371 CBA2D3 70692197 IC50 = 12.5 nM T20371 C0E5VQ 70692198 IC50 = 0.9 nM T20371 CRQ98X 70692199 IC50 = 5.7 nM T20371 C1WC7H 70693969 IC50 = 1950 nM T20371 CNL86O 70693988 IC50 = 7.8 nM T20371 CHKO91 70694038 IC50 = 4.9 nM T20371 CZ8WG6 70694039 IC50 = 0.9 nM T20371 CUNJ84 70694040 IC50 = 4.9 nM T20371 CM9GW7 70694041 IC50 = 73 nM T20371 C87MZC 70694042 IC50 = 11 nM T20371 CAK2R0 70696089 IC50 = 0.2 nM T20371 C4Z6KB 70696357 IC50 = 1.1 nM T20371 C1WL2C 71237709 IC50 = 30 nM T20371 C0NA8W 71238141 IC50 = 7 nM T20371 CV5X0O 71238209 IC50 = 300 nM T20371 CV4U6L 71238213 IC50 = 1000 nM T20371 CU0NH5 72546987 IC50 = 29 nM T20371 C5WXJ6 72546988 IC50 = 2.5 nM T20371 CBK6T9 72546989 IC50 = 1.2 nM T20371 C57QJB 72546990 IC50 = 440 nM T20371 C7C4HR 72547251 IC50 = 3 nM T20371 CY19IP 72547496 IC50 = 2.2 nM T20371 COF6E7 76313510 IC50 = 198 nM T20371 C42OQG 76327949 IC50 = 43 nM T20371 CWD5R4 76331595 IC50 = 2.5 nM T20371 C2H8OY 86276235 IC50 = 105 nM T20371 C92YAH 86276247 IC50 = 3.3 nM T20371 CIP5O9 90654431 IC50 = 270 nM T20371 CJ6A7G 90654433 IC50 = 10.4 nM T20371 C5B2ZG 90654435 IC50 = 74 nM T20371 C1B0XZ 90654436 IC50 = 3.5 nM T20371 C5AE6I 90654437 IC50 = 40 nM T20371 CET9X8 90654439 IC50 = 13 nM T20371 CH34UQ 90654440 IC50 = 69 nM T20371 C46RSL 90654441 IC50 = 40 nM T20371 CCF05S 90654442 IC50 = 66 nM T20371 C5QM6F 90654444 IC50 = 860 nM T20371 CP7T1E 90654446 IC50 = 940 nM T20371 CN3VO2 90654448 IC50 = 580 nM T20371 CW7OD5 90654450 IC50 = 990 nM T20371 CG6JB2 90654452 IC50 = 850 nM T20371 CBU5H8 90654454 IC50 = 92 nM T20371 C14JPC 90654456 IC50 = 114 nM T20371 CK19FW 90654457 IC50 = 150 nM T20371 CCE1O5 90654458 IC50 = 1500 nM T20371 C7ZBN6 90654459 IC50 = 150 nM T20371 D00VKV 62751 IC50 = 20 nM T20371 D09TDI 6472 Ki = 26 nM T20371 D0Q5PC 6468 IC50 = 91 nM T01003 D0E3TC 44259 IC50 = 204 nM T01003 D0AV6X 25160990 IC50 > 20000 nM T01003 CR5F4X 6195 IC50 > 20000 nM T01003 C12TIO 6998 IC50 > 20000 nM T01003 C9LD6W 7024 IC50 > 20000 nM T01003 C3ET2I 12819 IC50 = 9732 nM T01003 CV3O5S 16790 IC50 > 20000 nM T01003 CITN94 79352 IC50 > 20000 nM T01003 CHT53C 113099 IC50 > 20000 nM T01003 CD8J9V 11963346 IC50 > 50000 nM T01003 CMGU60 12934390 IC50 = 206 nM T01003 CB1MY8 60196244 IC50 = 290 nM T01003 CRX81Q 71575642 IC50 > 10000 nM T01003 CLTG58 78350466 IC50 = 14 nM T01003 C31OAQ 86290367 IC50 = 472 nM T01003 CLY3D1 86290407 IC50 = 296 nM T01003 CG6YQ8 86290408 IC50 = 181 nM T01003 CU1R5A 86290409 IC50 = 118 nM T01003 C0V5OB 86290410 IC50 = 111 nM T01003 C1VBT9 86290411 IC50 = 118 nM T01003 C8EXO1 86290412 IC50 = 150 nM T01003 CS75OW 86290413 IC50 > 20000 nM T01003 CO84KL 86290454 IC50 > 20000 nM T01003 CY2TV9 86290455 IC50 = 3051 nM T01003 CX32CK 86290456 IC50 > 20000 nM T01003 CP6M9F 86290457 IC50 > 20000 nM T01003 CXK21B 86290458 IC50 = 1230 nM T01003 CT4L8U 86290459 IC50 = 113 nM T01003 CGKV34 86290460 IC50 = 303 nM T01003 CE24CR 86290499 IC50 = 255 nM T01003 CS15PM 86290501 IC50 > 20000 nM T01003 C3V8DA 86290502 IC50 > 20000 nM T01003 C7CTJ6 86290503 IC50 > 20000 nM T01003 CJ81IB 86290504 IC50 = 1718 nM T01003 CUIK08 86290505 IC50 = 4109 nM T01003 CD16CO 86290541 IC50 = 5644 nM T01003 CWZ01E 86290542 IC50 > 20000 nM T01003 C17RVZ 86290569 IC50 = 200 nM T01003 CF47RW 86298445 IC50 = 312 nM T01003 CX4H6I 86583042 IC50 > 50000 nM T01003 CGAR65 90656471 IC50 > 20000 nM T01003 CE7TJ5 90656472 IC50 = 16210 nM T01003 CJ2NI1 118721229 IC50 = 71 nM T01003 CC05EY 118721230 IC50 = 14 nM T01003 C7HJ8Y 118721231 IC50 > 99000 nM T01003 C5XMF8 118721232 IC50 = 170 nM T01003 CZY01I 118721233 IC50 = 29 nM T01003 C2USQ7 118721234 IC50 = 51 nM T01003 CDS2U3 118721235 IC50 = 9.7 nM T01003 C0H9OV 118721236 IC50 = 11 nM T01003 C83KJY 118721237 IC50 = 6.4 nM T01003 C13QEP 118721238 IC50 = 5.1 nM T01003 CVC3B0 118721239 IC50 = 14 nM T01003 C2F6MN 118721240 IC50 = 45 nM T01003 C36PRN 118721241 IC50 = 54 nM T01003 CY0J8A 118721242 IC50 = 12 nM T01003 CJLX62 118721243 IC50 = 22 nM T01003 C14BFC 118721244 IC50 = 13 nM T01003 C6ETU2 118721245 IC50 = 31 nM T01003 C4TXF2 118730409 IC50 > 50000 nM T01003 C4X7SD 122192466 IC50 > 10000 nM T01003 CY28AI 135398515 IC50 = 9939 nM T01003 CKO83Y 136664429 EC50 = 143 nM T01003 CPC5O0 137333978 IC50 = 303 nM T01003 CA93HF 139593294 IC50 = 160 nM T01003 C2MD1Q 155513187 IC50 > 10000 nM T01003 CN47JC 155517517 IC50 = 72 nM T01003 C5U0SQ 155521969 IC50 = 130 nM T01003 C8N4OH 155522759 IC50 = 90 nM T01003 CRJF80 155525584 IC50 > 10000 nM T01003 CR51DL 155530872 IC50 > 10000 nM T01003 CN0PW5 155533307 IC50 = 190 nM T01003 CET2Q5 155539312 IC50 = 4060 nM T01003 C1TOM0 155540070 IC50 = 200 nM T01003 C1UM3W 155540082 IC50 = 100 nM T01003 C0RWS7 155542155 IC50 > 10000 nM T01003 CV6ZI7 155543519 IC50 > 10000 nM T01003 C5MHX7 155546098 IC50 = 130 nM T01003 CW4QJ2 155547079 IC50 = 110 nM T01003 CTZ5N8 155548986 IC50 = 160 nM T01003 CIR6U2 155551979 IC50 = 33 nM T01003 CY4P0U 155554101 IC50 = 890 nM T01003 CQH9K8 155555756 IC50 > 10000 nM T01003 CS5OW0 155560180 IC50 = 240 nM T01003 CFOP01 155560487 IC50 = 160 nM T01003 CE5W2A 155560538 IC50 = 2700 nM T01003 C8F6IT 155566735 IC50 = 840 nM T01003 D0E3CB 86290500 IC50 = 47 nM T01003 D0W1NH 72881 IC50 > 20000 nM T44387 D0E3TC 44259 IC50 = 3.8 nM T44387 D0O6WV 24794418 IC50 > 500 nM T44387 D03BNU 59604787 IC50 > 10000 nM T44387 CV63UL 67240318 IC50 > 10000 nM T44387 CPG3A5 86302574 IC50 > 30000 nM T44387 CUO0C5 132156633 IC50 > 10000 nM T44387 C2MD1Q 155513187 IC50 > 10000 nM T44387 D00ERW 44444843 Ki > 1650 nM T44387 D02NNT 53232451 IC50 = 224 nM T44387 D0E7VO 59627005 IC50 < 100 nM T14945 D0V2YJ 11655511 IC50 > 50000 nM T14945 C2FLZ8 65751 IC50 = 29600 nM T14945 CB5HD3 10554501 IC50 = 2100 nM T14945 CM08RL 71664472 EC50 = 79 nM T14945 C20TKN 71769545 IC50 = 100 nM T14945 C67TLF 71769546 IC50 = 8500 nM T14945 CW90VL 71769547 IC50 = 2100 nM T14945 C7QZC2 71769678 IC50 = 50 nM T14945 C8PE6L 71769679 IC50 = 1500 nM T14945 C8EMV1 71769680 IC50 = 1800 nM T14945 CO62BR 71769681 IC50 = 72 nM T14945 C7XQ9I 71769682 IC50 = 300 nM T14945 CSO09B 71769813 IC50 = 32 nM T14945 CP30XD 71769814 IC50 = 2000 nM T14945 C1HY6E 71769815 IC50 = 370 nM T14945 CB9W5R 71769816 IC50 = 35 nM T14945 CI1G7Z 71769817 IC50 = 140 nM T14945 CQU21O 71769935 IC50 = 540 nM T14945 C2W6VF 140271393 IC50 = 14 nM T14945 C3ES5B 140271434 IC50 = 19 nM T14945 CZ9JI7 155533484 IC50 = 2.2 nM T14945 CM10VF 155534465 IC50 = 1.5 nM T14945 CTZ41W 155540671 IC50 = 24 nM T14945 CK53JZ 155543498 IC50 = 1.7 nM T14945 CAD28R 155565238 IC50 = 1.6 nM T46482 D06CTE 57469 EC50 = 2120 nM T46482 D0OJ4L 3652 IC50 = 800 nM T46482 D08JWC 46241268 EC50 = 290 nM T46482 D0C8KF 159603 EC50 = 260.1 nM T46482 D0T1FC 10309114 EC50 = 2657 nM T46482 COQ02K 55658 EC50 = 107000 nM T46482 CW9OJ4 130714 EC50 = 95000 nM T46482 CEO4Y8 2741936 IC50 = 2880 nM T46482 CKD3J4 2744062 IC50 = 44800 nM T46482 C51UQV 2797476 IC50 = 1400 nM T46482 CCJ6A3 2809299 IC50 = 38000 nM T46482 CT62KM 7964426 IC50 = 17000 nM T46482 C5XCM8 7971597 IC50 = 24700 nM T46482 C4GB7J 9332337 IC50 = 17000 nM T46482 C1XSP6 9332820 IC50 = 22000 nM T46482 C0V8YD 9816506 EC50 = 829 nM T46482 CM35YR 9818270 EC50 = 63.7 nM T46482 C9RYX0 9930010 EC50 = 10.3 nM T46482 C7SR0H 10018576 EC50 = 399.4 nM T46482 C67RJK 10317115 EC50 = 51.5 nM T46482 CYX5L4 10359083 EC50 = 32 nM T46482 CI1VH7 11223759 EC50 = 108 nM T46482 CN9P5V 11558911 EC50 = 166 nM T46482 C8Q0GO 11596538 EC50 = 25.7 nM T46482 CYT12H 11647322 EC50 = 8.1 nM T46482 C1S7RJ 11695850 EC50 = 28.1 nM T46482 CXZ69V 11949605 EC50 = 5 nM T46482 CYU4Z2 13982892 EC50 = 955 nM T46482 CMQ9T0 16805564 EC50 = 15400 nM T46482 C09HXM 16876274 EC50 = 57400 nM T46482 C3HUO6 16876280 EC50 = 44000 nM T46482 C95HYG 20998392 EC50 = 8300 nM T46482 C0OC1K 20998396 EC50 = 10900 nM T46482 CBO10H 21003203 EC50 = 16800 nM T46482 C0TM6X 21470208 EC50 = 8.58 nM T46482 C01JYU 23079483 EC50 = 50.1 nM T46482 C5YT6P 23158703 EC50 = 312.3 nM T46482 CIG38J 23158770 EC50 = 187.9 nM T46482 C4KI0G 23158775 EC50 = 75 nM T46482 CYP14O 24513539 IC50 = 2400 nM T46482 CV9CZ4 24765332 EC50 = 102 nM T46482 CP1S4C 24860861 EC50 > 10000 nM T46482 CF6Y8K 24860863 EC50 = 4400 nM T46482 C72OMH 24860931 EC50 = 3200 nM T46482 CHY9G3 24898957 EC50 = 10 nM T46482 CV3AZ2 25070826 EC50 = 5.4 nM T46482 CHT7J5 25070827 EC50 = 48.5 nM T46482 C7YG6C 25070828 EC50 = 9.4 nM T46482 CV9S6P 25070829 EC50 = 72.8 nM T46482 CT4F8R 25070830 EC50 = 7.4 nM T46482 CPTF43 25071149 EC50 = 50.2 nM T46482 CX3RU1 25071150 EC50 = 15.2 nM T46482 C71AMU 25071151 EC50 = 7.2 nM T46482 CW3TB2 25154304 EC50 = 99 nM T46482 CJA48W 25650103 EC50 = 6300 nM T46482 CM9AC5 26273315 IC50 = 3900 nM T46482 C13AWM 26718455 IC50 = 4400 nM T46482 CC2I4U 27661906 IC50 = 15000 nM T46482 CXWQ58 27662121 IC50 = 1830 nM T46482 CI5N7W 27662197 IC50 = 3090 nM T46482 C8IYP2 27662233 IC50 = 2100 nM T46482 CSL0G9 42606777 EC50 = 474 nM T46482 C4E0XK 42613092 IC50 = 25000 nM T46482 CO5WD1 44138041 IC50 = 7500 nM T46482 CV2RB0 44415366 EC50 = 790 nM T46482 CRS47C 44588952 EC50 = 100 nM T46482 C0N3AL 44588973 EC50 = 10 nM T46482 CHXE50 44588974 EC50 < 20 nM T46482 CGT9A6 44588975 EC50 < 20 nM T46482 CYCQ23 44592365 IC50 = 0.65 ug.mL-1 T46482 C9STJ2 44592366 EC50 = 2000 nM T46482 CQAJ97 45102599 IC50 = 1990 nM T46482 C2P0DG 46196912 EC50 = 609.1 nM T46482 C7CO0L 46196913 EC50 = 72.9 nM T46482 C4TAF6 46196914 EC50 = 466.8 nM T46482 CDHL70 46196915 EC50 = 87.5 nM T46482 CMFD53 46523001 IC50 = 5800 nM T46482 C8HVW3 46830487 EC50 = 472 nM T46482 C37FOD 46830488 EC50 = 647 nM T46482 C04MCE 46830489 EC50 = 59.1 nM T46482 COL8P4 46830776 EC50 = 91.5 nM T46482 CC0DK5 46830777 EC50 = 479 nM T46482 CYLP38 46830778 EC50 = 822 nM T46482 CFG82B 46830779 EC50 = 3350 nM T46482 C1YNK2 46831065 EC50 = 262 nM T46482 C5AH2C 46831067 EC50 = 209 nM T46482 C5DIS6 46831372 EC50 = 723 nM T46482 CC32AL 46831374 EC50 = 873 nM T46482 C84UPC 46831378 EC50 = 385 nM T46482 CHBX40 46834248 EC50 = 7710 nM T46482 CQ06VW 46834530 EC50 = 8390 nM T46482 CZ03LQ 47445274 IC50 = 30000 nM T46482 CXV2J0 49771644 EC50 = 1540 nM T46482 CF40TR 49771645 EC50 = 266 nM T46482 CAQ1Y3 49771648 EC50 = 100 nM T46482 C8AM4S 49771650 EC50 = 50 nM T46482 CL4XV5 49771651 EC50 = 87 nM T46482 CE2VI3 49771655 EC50 = 480 nM T46482 C40XQI 49771656 EC50 = 304 nM T46482 C2Y6AR 49771669 EC50 > 4000 nM T46482 CKO32M 49771672 EC50 = 1440 nM T46482 CR2PB7 49838133 EC50 = 310 nM T46482 C3AN6Q 49838134 EC50 = 240 nM T46482 CH6YV3 49838260 EC50 = 350 nM T46482 CN10ZM 49838385 EC50 = 390 nM T46482 C2N0FR 49838386 EC50 = 150 nM T46482 CB2JH7 49838387 EC50 = 90 nM T46482 C2F3OT 49838509 EC50 = 200 nM T46482 C1R8CE 49838511 EC50 = 5600 nM T46482 CRW6D9 49838512 EC50 = 65 nM T46482 C2XM1C 49838641 EC50 = 39 nM T46482 C3L2MV 49838771 EC50 = 980 nM T46482 C5JBY1 49838772 EC50 = 3100 nM T46482 CA2MP4 50899555 EC50 = 247 nM T46482 C0G6OM 51204571 IC50 = 1000 nM T46482 CZB84N 52941850 EC50 = 396 nM T46482 C8OK9G 52944297 EC50 = 110 nM T46482 C3PU5J 52945312 EC50 = 20 nM T46482 C1N9QU 52946707 EC50 = 396 nM T46482 CA3DJ6 52946880 EC50 = 108 nM T46482 C4JS7O 52948094 EC50 = 115 nM T46482 CQ24EO 53257973 IC50 = 820 nM T46482 C2QN7J 53257974 IC50 = 8580 nM T46482 C9UD7J 53257975 IC50 = 14850 nM T46482 C1XQM2 53484134 EC50 = 2.7 nM T46482 CTH2E7 54581014 EC50 = 411 nM T46482 C8MEA6 54582996 EC50 = 352 nM T46482 C1J5DU 54583999 EC50 = 95 nM T46482 CX0CL6 54584665 EC50 = 269 nM T46482 CF0U6X 54584939 EC50 = 193 nM T46482 C2BOV8 54584981 EC50 = 633 nM T46482 CKN5X6 54584982 EC50 > 4000 nM T46482 CAF6Q7 54585905 EC50 = 103 nM T46482 CW5TD8 54585906 EC50 = 79 nM T46482 C6UMY3 54585937 EC50 = 51 nM T46482 C6XBK5 54585938 EC50 > 4000 nM T46482 C38OAR 54586596 EC50 = 2200 nM T46482 C36IQE 54586874 EC50 = 833 nM T46482 C2G8LD 54586875 EC50 = 328 nM T46482 CG8F7K 54586876 EC50 = 366 nM T46482 C9CY4L 54760856 IC50 > 970 nM T46482 C9KSY0 56658701 EC50 = 9 nM T46482 CJN13I 56658873 EC50 = 2.3 nM T46482 C58JEI 56659528 IC50 = 38730 nM T46482 CD4LS6 56659557 IC50 = 22040 nM T46482 CJHY21 56659558 IC50 = 10140 nM T46482 CP72FK 56662183 EC50 = 2.7 nM T46482 C2HY7M 56662357 EC50 = 121 nM T46482 CE9H3A 56663006 IC50 = 19900 nM T46482 C21DRJ 56663007 IC50 = 21120 nM T46482 CKU56Y 56665640 EC50 = 1.7 nM T46482 C8ROD6 56665641 EC50 = 26.9 nM T46482 C7EKA9 56665642 EC50 = 6.6 nM T46482 CA56BG 56665643 EC50 = 1.5 nM T46482 C2TJV4 56665644 EC50 = 1.6 nM T46482 CFZD24 56665787 EC50 = 1780 nM T46482 C08RFC 56665788 EC50 = 2610 nM T46482 C24OXU 56665789 EC50 = 105 nM T46482 CRA47V 56666449 IC50 = 46500 nM T46482 C0P2LQ 56666450 IC50 = 26100 nM T46482 CLIE90 56666451 IC50 = 30440 nM T46482 C63AVI 56666452 IC50 = 37240 nM T46482 CRJ08Q 56666485 IC50 = 14400 nM T46482 CJ5TQ0 56666486 IC50 = 46400 nM T46482 CFWV74 56666487 IC50 = 4810 nM T46482 CC82PN 56669090 EC50 = 0.2 nM T46482 CG37WP 56669245 EC50 = 125 nM T46482 CT5YD1 56669246 EC50 = 47 nM T46482 CKPE85 56669899 IC50 = 20320 nM T46482 C41FRT 56672554 EC50 = 6.6 nM T46482 CDAR19 56672555 EC50 = 4.1 nM T46482 CXK31N 56672556 EC50 = 1 nM T46482 C0S2CF 56672557 EC50 = 0.4 nM T46482 CR9QO8 56672558 EC50 = 31 nM T46482 CT28HF 56672711 EC50 = 81.9 nM T46482 C8YEB4 56672712 EC50 = 45.8 nM T46482 CC8IN0 56673358 IC50 = 28020 nM T46482 CBWT27 56675929 EC50 = 121 nM T46482 CXYE78 56676070 EC50 = 920 nM T46482 CAX7T5 56679241 EC50 = 6.9 nM T46482 C1BJ7P 56679242 EC50 = 1.7 nM T46482 CA9L2D 56680005 IC50 = 38420 nM T46482 CUSG48 56682558 EC50 = 32.1 nM T46482 C4ED0Q 56682695 EC50 = 586 nM T46482 CD9NT0 56682696 EC50 = 55.4 nM T46482 CY8I7H 56682697 EC50 = 28.6 nM T46482 C0D4UI 56683347 IC50 = 21170 nM T46482 CGV53C 56683348 IC50 = 21630 nM T46482 CV2R1D 56954508 IC50 = 50 nM T46482 CD63TK 56954511 IC50 = 17880 nM T46482 CXC7H6 56954615 IC50 = 2050 nM T46482 C4HP7Y 56954616 IC50 = 560 nM T46482 C59AFV 56954617 IC50 = 3000 nM T46482 CDL64W 56954728 IC50 = 1420 nM T46482 C6AU7V 56954729 IC50 = 110 nM T46482 C5OZ7U 56954730 IC50 = 240 nM T46482 CN37MX 56954731 IC50 = 560 nM T46482 C7ZR3S 56954831 IC50 = 170 nM T46482 CUL8K7 56954832 IC50 = 450 nM T46482 C8M9XY 56954833 IC50 = 7240 nM T46482 CH9X0M 56954948 IC50 = 4020 nM T46482 CR0QZ6 56954949 IC50 = 5400 nM T46482 C23XPA 58166514 EC50 = 230 nM T46482 CCHP08 59252568 EC50 = 2600 nM T46482 C6E4IV 59281148 EC50 = 19.6 nM T46482 CV72GW 67181623 EC50 = 150 nM T46482 CK2V9S 67182494 EC50 = 100 nM T46482 C8P9WA 67183000 EC50 = 230 nM T46482 C1JC6H 67183672 EC50 = 900 nM T46482 CMO74J 67185919 EC50 = 620 nM T46482 CZ1DF2 67607124 EC50 = 3950 nM T46482 CDCT67 68322071 EC50 = 150 nM T46482 CIQ29G 70703181 EC50 = 4000 nM T46482 CH29GF 71258526 IC50 > 10000 nM T46482 CR9AY7 71284052 EC50 = 1200 nM T46482 C54YUS 71292238 EC50 > 270000 nM T46482 C61EPX 71292267 EC50 = 4400 nM T46482 CXQ26G 71292269 EC50 = 2900 nM T46482 CS4AF1 71292276 EC50 = 14370 nM T46482 CR6QJ7 71292278 EC50 = 2220 nM T46482 CN4E2D 71292284 EC50 = 49200 nM T46482 CWA83L 71292294 EC50 = 29100 nM T46482 CG8Z6Y 71292304 EC50 = 5700 nM T46482 C8GNX0 71292306 EC50 = 4800 nM T46482 CMR0W9 71505363 EC50 = 2600 nM T46482 CWB56Z 71505551 EC50 = 2420 nM T46482 CG29QY 71505730 EC50 = 23800 nM T46482 CQMT93 71520574 EC50 = 165.7 nM T46482 CCE05D 71717369 EC50 = 9.3 nM T46482 CN0K7D 71717370 EC50 = 7.6 nM T46482 CGD60L 71717965 EC50 = 30.1 nM T46482 C5W9VU 71719186 EC50 = 7 nM T46482 CRGM24 71719187 EC50 = 130 nM T46482 CTX54P 71719791 EC50 = 58 nM T46482 C6DF0Q 71899933 EC50 = 66600 nM T46482 C8XO4L 73774707 EC50 = 100 nM T46482 CNY9K2 73774844 EC50 = 9 nM T46482 CI7J8R 73775160 EC50 = 140 nM T46482 C28OEA 73775161 EC50 = 90 nM T46482 CMXZ65 86346192 EC50 = 61 nM T46482 CN6OU1 90668083 EC50 > 4000 nM T46482 CD6SI2 90668084 EC50 > 4000 nM T46482 C1BPN5 90668085 EC50 > 4000 nM T46482 CG6U3J 90668086 EC50 > 4000 nM T46482 CG7H8A 90668087 EC50 > 4000 nM T46482 CM4AB1 90668088 EC50 > 4000 nM T46482 C0PKF2 90668089 EC50 > 4000 nM T46482 CN1DP8 90668090 EC50 > 4000 nM T46482 CMH6I5 90668091 EC50 > 4000 nM T46482 CN01DH 117886834 EC50 = 60 nM T46482 CO5CD6 117886835 EC50 = 60 nM T46482 C4K2EH 117886860 EC50 = 260 nM T46482 C6XS8J 117887024 EC50 = 1 nM T46482 CP0I7M 117887098 EC50 = 6 nM T46482 C02WMX 117887431 EC50 = 30 nM T46482 CIF48S 117887482 EC50 = 220 nM T46482 CGQK61 117887492 EC50 = 280 nM T46482 C6H8TA 117887507 EC50 = 60 nM T46482 CA7Z3W 117887511 EC50 = 6 nM T46482 CFV23K 117887619 EC50 = 0.6 nM T46482 CBR40O 117887688 EC50 = 40 nM T46482 CB0ZR1 117887696 EC50 = 750 nM T46482 C82IKQ 117887700 EC50 = 420 nM T46482 C1B4EZ 117887727 EC50 < 10 nM T46482 C1NBR2 118334961 EC50 < 10 nM T46482 C6HJY4 118334964 EC50 = 130 nM T46482 CF7V8I 118334970 EC50 = 2200 nM T46482 CKG4L3 118334971 EC50 = 9 nM T46482 CRV14T 118334974 EC50 = 30 nM T46482 C7VYK2 118334975 EC50 = 8 nM T46482 CZ36OR 118334976 EC50 = 20 nM T46482 CR8U2Y 118334978 EC50 = 500 nM T46482 CIS2L9 118334979 EC50 = 9 nM T46482 CJS5E1 118334980 EC50 = 20 nM T46482 CKM6L0 118334982 EC50 = 40 nM T46482 C0ZF5S 118334989 EC50 = 50 nM T46482 C0SVW4 118334990 EC50 = 130 nM T46482 CH8PU2 118334995 EC50 = 20 nM T46482 CO3PU6 118334997 EC50 = 2200 nM T46482 CTUO62 118334999 EC50 = 1000 nM T46482 C8EBN6 118335005 EC50 = 560 nM T46482 CEBR65 118335006 EC50 = 500 nM T46482 C4T3XE 118335013 EC50 = 70 nM T46482 CU4E5M 118335014 EC50 = 40 nM T46482 CZO7F9 118335018 EC50 = 130 nM T46482 CM78SL 118335021 EC50 = 6 nM T46482 CK83OB 118335025 EC50 = 150 nM T46482 C7IU8N 121401335 EC50 = 1960 nM T46482 C7NWK8 121401336 EC50 = 99 nM T46482 C5RXG7 121401340 EC50 = 100 nM T46482 CV0FH9 121401343 EC50 = 6 nM T46482 CAE1L7 130289620 EC50 = 2890 nM T46482 CF5LT4 130289627 EC50 = 4530 nM T46482 CBI4C0 130289680 EC50 = 190000 nM T46482 C71EHG 130289685 EC50 = 1740 nM T46482 C2BA3W 130289686 EC50 = 2890 nM T46482 CJH93E 130289687 EC50 = 180 nM T46482 CJY9E3 130289827 EC50 = 600 nM T46482 CVWZ36 130289832 EC50 = 3330 nM T46482 CE8KQ3 130289845 EC50 = 3840 nM T46482 C4EJQ0 130289846 EC50 = 6670 nM T46482 CK86LY 130290425 EC50 = 3060 nM T46482 CXN30J 130290443 EC50 = 3640 nM T46482 C6NTM8 130454358 IC50 = 1400 nM T46482 C59JSA 130454361 IC50 = 17000 nM T46482 C26WUT 130454401 IC50 = 11000 nM T46482 C6FHY8 130454431 IC50 = 700 nM T46482 C6B9XI 130454445 IC50 = 53000 nM T46482 CIU01F 130454450 IC50 = 1200 nM T46482 CHAE81 130454459 IC50 = 31000 nM T46482 CVEF58 130454467 IC50 = 52000 nM T46482 CG08CU 130454481 IC50 = 5600 nM T46482 CTOG04 130454512 IC50 = 1300 nM T46482 CY4JT1 130454516 IC50 = 4400 nM T46482 C8RUV4 130454546 IC50 = 16000 nM T46482 C7JNE6 130454574 IC50 = 4900 nM T46482 CF06GU 130454579 IC50 = 20700 nM T46482 CBM73C 130454634 IC50 = 1200 nM T46482 CXNZ71 130454680 IC50 = 9600 nM T46482 CE86DQ 130454681 IC50 = 4600 nM T46482 C0U4FJ 130472372 IC50 = 17000 nM T46482 CI84KG 130472422 IC50 = 5800 nM T46482 C93TUC 130472439 IC50 = 1400 nM T46482 C28LWH 130472440 IC50 = 8700 nM T46482 C45BQH 132585194 EC50 > 100000 nM T46482 CBC87Y 134229125 IC50 > 20000 nM T46482 C2DO5I 134229163 IC50 < 1000 nM T46482 C79HWU 134229173 IC50 < 1000 nM T46482 C2N7FJ 134229210 IC50 < 1000 nM T46482 CR2LC4 134229258 IC50 < 1000 nM T46482 CB3JV5 134229300 IC50 < 1000 nM T46482 C2B5HY 134229340 IC50 < 1000 nM T46482 C37BCL 134237203 IC50 < 1000 nM T46482 CL3PN6 134237231 IC50 < 1000 nM T46482 C9WYC1 134237255 IC50 < 1000 nM T46482 C76FIZ 134242384 IC50 = 1000 nM T46482 C7WG8O 135260399 EC50 = 1020 nM T46482 C15GPU 135260404 EC50 = 3260 nM T46482 C0OC5M 135260416 EC50 = 2890 nM T46482 CC8SJ4 135260424 EC50 = 1290 nM T46482 C96OZB 135260428 EC50 = 398 nM T46482 C02NFK 135271001 EC50 = 3400 nM T46482 CF1J7O 135271003 EC50 = 590 nM T46482 C2JXW8 135271007 EC50 = 510 nM T46482 CGD0Y6 135271008 EC50 = 730 nM T46482 COC2D9 135271011 EC50 = 1270 nM T46482 C6KGY3 135271012 EC50 = 958 nM T46482 CRE58J 135271014 EC50 = 46 nM T46482 CF8AX4 135271016 EC50 = 379 nM T46482 C4LX5U 135271017 EC50 = 375 nM T46482 COL31X 135271018 EC50 = 1240 nM T46482 CG6Y7B 135271021 EC50 = 1100 nM T46482 CK5FB8 135271028 EC50 = 710 nM T46482 CWG6U8 135271030 EC50 = 140 nM T46482 CB6J0X 135271031 EC50 = 1160 nM T46482 CTSI07 135271032 EC50 = 262 nM T46482 CWL20P 135271033 EC50 = 714 nM T46482 C29UTE 135271034 EC50 = 1160 nM T46482 C5N3YE 135271038 EC50 = 562 nM T46482 CB3G8N 135271039 EC50 = 1400 nM T46482 CJDE91 135271042 EC50 = 265 nM T46482 CO7CT1 135271043 EC50 = 194 nM T46482 CC2S6G 135271044 EC50 = 2820 nM T46482 CE0F5R 135271045 EC50 = 251 nM T46482 C8UBG3 137515213 EC50 > 100000 nM T46482 C5Q6TS 137515380 EC50 > 100000 nM T46482 CNT8G1 137515383 EC50 > 100000 nM T46482 CVI1H4 137515466 EC50 > 100000 nM T46482 CKC32Q 137515546 EC50 > 100000 nM T46482 C6Q5YE 137515571 EC50 > 100000 nM T46482 CJ85ER 137515794 EC50 > 100000 nM T46482 CSU98Z 137515846 EC50 > 100000 nM T46482 C0M6SU 137515935 EC50 > 100000 nM T46482 C4TGP3 137516041 EC50 > 100000 nM T46482 CS15BK 137516054 EC50 > 100000 nM T46482 C0F5XW 137516341 EC50 > 100000 nM T46482 C1DQ9N 137632868 IC50 = 4990 nM T46482 C6UK4P 137640101 IC50 = 10840 nM T46482 C5UP7W 137640859 IC50 = 8300 nM T46482 CN4T8D 137644178 IC50 = 7550 nM T46482 CUIL14 137645168 IC50 = 66170 nM T46482 CQ0A7B 137647183 IC50 = 4570 nM T46482 C0O6SE 137658022 EC50 = 1640 nM T46482 CXZL91 137661216 IC50 = 4710 nM T46482 CSUN37 137661892 IC50 = 8090 nM T46482 CH1JE8 138605929 EC50 = 3210 nM T46482 C0B7CD 138605940 EC50 = 1720 nM T46482 CL9YN6 139030521 IC50 = 8200 nM T46482 C7RM0D 145964333 IC50 = 27000 nM T46482 CGK05C 145965353 IC50 = 260 nM T46482 CV54KR 145966301 IC50 = 14000 nM T46482 CFS9C3 145966325 IC50 = 23200 nM T46482 C2UZE8 145967009 IC50 = 27800 nM T46482 CG47YZ 145967371 IC50 = 25000 nM T46482 CUHS36 145969404 IC50 = 500 nM T46482 CU20BN 145969832 IC50 = 2600 nM T46482 C2EJ6H 145970777 IC50 = 17260 nM T46482 C3UK8W 145970984 IC50 = 13400 nM T46482 C9UG6K 145972030 IC50 = 1900 nM T46482 CT9FH0 145974655 IC50 = 16000 nM T46482 CO6D0K 145975440 IC50 = 60000 nM T46482 C5F6GX 145975659 IC50 = 440 nM T46482 CW3N6D 145976358 IC50 = 990 nM T46482 CH5RZ9 145977142 IC50 = 7900 nM T46482 C8JS6I 145977414 IC50 = 1020 nM T46482 C4FAZ7 145978184 IC50 = 14200 nM T46482 CH4LN3 145978832 IC50 = 900 nM T46482 CWZ59N 145978968 IC50 = 4200 nM T46482 C9K6JX 145983197 IC50 < 1000 nM T46482 CGVS82 145986851 IC50 = 5700 nM T46482 C6TV1L 145988217 IC50 = 11000 nM T46482 CZ2HG1 145989953 IC50 = 22000 nM T46482 C6BMI0 145990319 IC50 = 5400 nM T46482 CDQP96 145992257 IC50 = 17000 nM T46482 CNS1C9 145998100 IC50 = 10000 nM T46482 C6L8VP 145998103 IC50 = 17300 nM T46482 C86ZCE 145998104 IC50 = 22000 nM T46482 CG21HD 145998105 IC50 = 17700 nM T46482 CT81ZB 154734323 IC50 > 50000 nM T46482 CV4RP7 154734324 IC50 > 20000 nM T46482 C8I9WN 155510395 EC50 = 535000 nM T46482 C4HG5W 155510901 IC50 = 2650 nM T46482 CS59AL 155511147 IC50 > 50000 nM T46482 CM8A2L 155512278 IC50 = 39300 nM T46482 CFXE54 155513812 IC50 = 26000 nM T46482 CWT86N 155517386 IC50 = 43100 nM T46482 CCLH62 155519934 EC50 = 279000 nM T46482 CZV2X5 155520111 IC50 = 7100 nM T46482 C37YVX 155520248 EC50 = 4400 nM T46482 CS8B5U 155522619 IC50 = 15800 nM T46482 C60JPG 155522765 IC50 = 40000 nM T46482 CL8MA9 155525358 EC50 = 1800 nM T46482 C35WAO 155526329 IC50 > 50000 nM T46482 CAI94F 155527796 IC50 > 50000 nM T46482 CP14CH 155528952 IC50 = 48300 nM T46482 CKN85X 155529119 IC50 = 49500 nM T46482 CE9DF0 155529356 IC50 = 84000 nM T46482 CWG5Q4 155529545 IC50 > 50000 nM T46482 CGO36X 155529770 EC50 = 114000 nM T46482 CBLY37 155531175 IC50 = 6200 nM T46482 C8U0PK 155531703 IC50 > 50000 nM T46482 CBA05R 155532062 IC50 = 50000 nM T46482 C7C1FH 155532740 IC50 = 45000 nM T46482 CF35AP 155533240 IC50 = 2900 nM T46482 C8MWT1 155533267 IC50 = 23900 nM T46482 CJHS17 155534690 IC50 = 42500 nM T46482 C4OJ7I 155535320 IC50 = 16300 nM T46482 C81ONH 155536356 IC50 = 30600 nM T46482 C3IB9T 155536360 IC50 = 23500 nM T46482 CH9WQ6 155537812 IC50 > 50000 nM T46482 CUB76Z 155540600 IC50 = 4730 nM T46482 C0YQA5 155549325 IC50 = 42500 nM T46482 CLHW81 155551508 IC50 = 4700 nM T46482 C94SVT 155553856 IC50 = 39000 nM T46482 CFJ78Q 155554706 EC50 = 29900 nM T46482 C1AZ9I 155555126 IC50 = 40000 nM T46482 CT79FB 155556399 IC50 = 1000 nM T46482 C7IH5O 155557699 IC50 = 25000 nM T46482 CIKL52 155559456 IC50 = 23600 nM T46482 C1D6TV 155560469 IC50 = 32500 nM T46482 CK5C3Z 155561314 IC50 > 50000 nM T46482 CB98NZ 155563615 IC50 > 50000 nM T46482 CMLJ58 155567376 IC50 = 48500 nM T46482 C90WLT 155568067 EC50 = 15000 nM T23785 C3VRO9 44557921 IC50 > 10000 nM T23785 C86YRV 58688296 IC50 > 30000 nM T23785 C8AT5N 58688313 IC50 > 30000 nM T23785 C09YWX 58688317 IC50 > 12500 nM T23785 C4Q2HL 58688342 IC50 = 2740 nM T23785 C0LK4S 58688380 IC50 > 30000 nM T23785 CNVK41 58688409 IC50 > 30000 nM T23785 CJI0Q4 58688436 IC50 > 30000 nM T23785 CZ0J6F 58688467 IC50 > 30000 nM T23785 CPE98M 58688474 IC50 > 30000 nM T23785 CDOK25 58688484 IC50 > 30000 nM T23785 CHO5G0 58688561 IC50 > 30000 nM T23785 CP2JK1 58688569 IC50 = 2013 nM T23785 CIV53P 58688575 IC50 = 415 nM T23785 C2T8UL 58688642 IC50 > 30000 nM T23785 CIJ5L9 70682556 IC50 > 30000 nM T23785 C9IB8C 70684645 IC50 = 612 nM T23785 CH08ZN 70690951 IC50 > 30000 nM T23785 CK0CH3 70697188 IC50 > 30000 nM T23785 C3B4HT 136003186 IC50 > 30000 nM T23785 D0F6NZ 58688690 IC50 = 415 nM T23785 D0FC4Y 46192505 IC50 = 252 nM T23785 D0S0XD 58688563 IC50 > 30000 nM T20776 CT0U8L 9815029 IC50 > 100000 nM T20776 C2P9NE 9858287 IC50 = 53800 nM T20776 C60IAQ 58619539 IC50 = 26900 nM T20776 CQSU96 91668553 IC50 = 1480 nM T20776 CGDW51 91668554 IC50 = 159 nM T20776 C1BX7Z 91668556 IC50 = 63200 nM T20776 C9LM8K 91668557 IC50 = 818 nM T20776 CF0MU1 118735141 IC50 = 6150 nM T20776 CPR4H8 118735142 IC50 = 141 nM T20776 C1F8YJ 118735143 IC50 = 190 nM T20776 C7V3SG 118735144 IC50 > 100000 nM T20776 CU07TA 118735145 IC50 = 1450 nM T20776 CS1WQ8 118735769 IC50 = 384 nM T20776 CFC42D 118735770 IC50 = 9180 nM T20776 CMHZ30 118735771 IC50 = 21100 nM T20776 CSB1V0 118735772 IC50 > 100000 nM T20776 CXN4E3 118735773 IC50 = 2520 nM T20776 C3OYE2 118735774 IC50 = 6840 nM T20776 C5U6TN 118735775 IC50 = 22800 nM T20776 CB1TD9 118735776 IC50 = 24890 nM T20776 C8TM3X 118735777 IC50 = 76100 nM T20776 CES82L 118735778 IC50 = 1820 nM T20776 CJDN52 118735779 IC50 > 100000 nM T20776 C7WM8V 118735780 IC50 = 76500 nM T20776 CBAN54 118735782 IC50 = 22000 nM T20776 C78XED 118735783 IC50 > 23700 nM T20776 CZOI63 118735784 IC50 = 2350 nM T20776 CF5RS3 118735785 IC50 > 100000 nM T20776 CQTH95 118735786 IC50 = 429 nM T20776 CO46US 118735787 IC50 = 374 nM T20776 CEA1Q3 118735788 IC50 = 108 nM T20776 CQ3ZF9 118735789 IC50 = 188 nM T20776 CUS6C9 118735790 IC50 = 15 nM T20776 CPF65J 118735791 IC50 = 25 nM T20776 CK4XS8 118735793 IC50 = 3570 nM T94131 D09XZB 123631 IC50 > 50000 nM T94131 D0B3HD 2519 IC50 = 1000000 nM T94131 D0E3SH 6918837 IC50 > 10000 nM T94131 D0E6XR 3062316 IC50 > 50000 nM T94131 D0F8RA 2153 IC50 = 800000 nM T94131 D0J5VR 11625818 IC50 = 60 nM T94131 D0K8KX 5280343 IC50 = 13790 nM T94131 D0R0MW 5329102 IC50 = 13000 nM T94131 D0RU0O 50905713 IC50 = 2 nM T94131 D0S5LD 135565596 IC50 = 0.7 nM T94131 D0W5HK 216239 IC50 > 50000 nM T94131 D01PGR 16123056 IC50 = 9 nM T94131 D01QSO 16654980 IC50 = 256 nM T94131 D03BHZ 52913813 IC50 = 675 nM T94131 D03EZE 25167777 IC50 = 0.61 nM T94131 D03FOP 68947304 IC50 = 850 nM T94131 D03IJO 11618268 IC50 = 3000 nM T94131 D03KAC 1893730 IC50 = 23 nM T94131 D03XAQ 49784945 IC50 = 36 nM T94131 D06GUA 49784002 IC50 = 6309.57 nM T94131 D07EHV 44814409 IC50 > 9100 nM T94131 D07HPJ 11476171 IC50 = 3200 nM T94131 D08QGT 17755052 Ki = 1.4 nM T94131 D0C3ZR 10427712 IC50 = 83 nM T94131 D0D8JB 44516953 IC50 = 6 nM T94131 D0E6UZ 54575456 IC50 = 311 nM T94131 D0I3LO 91933883 IC50 = 0.29 nM T94131 D0LG7X 86291103 IC50 = 33 nM T94131 D0O1LD 11647372 IC50 = 5 nM T94131 D0O6VZ 25254071 IC50 = 14 nM T94131 D0O8SJ 72950888 IC50 > 120 nM T94131 D0TU7B 58507717 IC50 = 708 nM T94131 D0U3DP 46912230 IC50 = 25 nM T94131 D0UP1Z 51001932 Ki = 0.97 nM T94131 D0VG0D 11977753 IC50 = 6 nM T94131 D0W7HE 56649450 IC50 = 250 nM T94131 D0X7IN 11978790 IC50 = 38 nM T94131 D0XD4I 118502708 IC50 = 1100 nM T94131 D0Y2NS 70798655 IC50 = 1900 nM T94131 D03BNU 59604787 IC50 > 5000 nM T94131 D0C9JZ 58111426 IC50 = 2297 nM T94131 D05HIJ 135565159 IC50 = 10000 nM T94131 D09SFV 3973 IC50 = 950 nM T94131 D0D0QA 44137675 IC50 = 1090 nM T94131 D0P1JI 312145 IC50 = 19 nM T94131 CX74ND 40237 IC50 = 380000 nM T94131 CEL9D8 79972 IC50 = 1498000 nM T94131 CNW59X 95001 IC50 = 53000 nM T94131 C3FRX9 131989 IC50 > 83300 nM T94131 C1MOD6 165595 IC50 = 2415000 nM T94131 CW1B9X 226105 IC50 = 1570000 nM T94131 C6KL2D 235602 IC50 = 992000 nM T94131 C4I2PT 244740 IC50 = 134000 nM T94131 C6ET7X 247414 IC50 = 5184000 nM T94131 CGC10Q 249363 IC50 = 2700 nM T94131 CQ7B2K 252311 IC50 = 187000 nM T94131 CBY29G 260801 IC50 = 105000 nM T94131 C1Y0JB 263480 IC50 = 324000 nM T94131 CTU12Q 267310 IC50 > 1600000 nM T94131 CJ43OR 270557 IC50 = 6074000 nM T94131 CV8DJ6 274101 IC50 = 241000 nM T94131 C2M5YF 275065 IC50 = 1460000 nM T94131 CEW10F 291727 IC50 = 234000 nM T94131 C1M3IR 309591 IC50 = 9157000 nM T94131 C6E4HJ 347279 IC50 = 5876000 nM T94131 CFW2K4 414938 IC50 = 2437000 nM T94131 COE1I6 426449 IC50 = 7333000 nM T94131 CK30NI 520127 IC50 > 1670000 nM T94131 CY3D4G 617191 IC50 = 16670 nM T94131 CS5O7B 622000 IC50 > 40000 nM T94131 CXC3V1 622262 IC50 = 1660 nM T94131 CU73NO 736009 IC50 > 83300 nM T94131 CZN6S9 743974 IC50 > 25118.86 nM T94131 C3P4OY 1093514 IC50 = 27950 nM T94131 C3KPX5 1270546 IC50 = 920 nM T94131 CP0QU1 1355022 IC50 = 3600 nM T94131 CWOQ49 1627922 IC50 = 10000 nM T94131 CAN89K 2762479 IC50 > 100000 nM T94131 C56YDF 2762944 IC50 > 100000 nM T94131 C8E3HY 2796894 IC50 = 5495.41 nM T94131 C09VKD 2816900 IC50 > 83300 nM T94131 C4RH3J 3106064 IC50 = 25000 nM T94131 C4PQ7T 3128427 IC50 = 5 nM T94131 C1O4KS 4416330 IC50 = 4200 nM T94131 CIN5F7 4904109 IC50 <= 10000 nM T94131 C1YJM9 4912089 IC50 > 83300 nM T94131 CE74CV 5059890 IC50 = 100000 nM T94131 C9N4MH 5765281 IC50 = 20000 nM T94131 CKX0F4 5806797 IC50 = 4300 nM T94131 C8CL1W 6053578 IC50 = 612000 nM T94131 CS26IV 6089668 IC50 = 3800 nM T94131 CGF7R0 6196488 IC50 = 20000 nM T94131 C2OZ0W 6484194 IC50 > 83300 nM T94131 CK2IR4 6852165 IC50 = 2030 nM T94131 CX18LU 9342140 IC50 = 1200 nM T94131 CE1Y8A 9815659 IC50 = 37000 nM T94131 CJ79RC 9879653 IC50 = 31 nM T94131 CC2Q6T 9925404 IC50 = 217800 nM T94131 CLT13A 10088066 IC50 = 4000 nM T94131 C9HWF6 10114067 IC50 = 3630 nM T94131 C57FPB 10115147 IC50 = 5450 nM T94131 CZ15SC 10125446 IC50 = 380 nM T94131 C02SQE 10141582 IC50 = 7620 nM T94131 CZ4D7S 10181657 IC50 = 145200 nM T94131 CF6Y2U 10202973 IC50 = 1820 nM T94131 C1RDW9 10203280 IC50 = 6170 nM T94131 CC82QV 10204538 IC50 = 137900 nM T94131 CO5VP9 10296641 IC50 = 2540 nM T94131 C7SFI1 10296883 IC50 > 10000 nM T94131 C7ZG0A 10296917 IC50 = 13070 nM T94131 CW7Q0R 10315189 IC50 = 18150 nM T94131 C32NQS 10357196 IC50 = 21 nM T94131 CC67FL 10383101 IC50 = 46000 nM T94131 C2VG4L 10455817 IC50 = 2.42 nM T94131 CAZT53 10475366 IC50 = 570 nM T94131 CL8YE3 11230964 IC50 = 6400 nM T94131 C8Y6IM 11234514 IC50 = 67 nM T94131 CK65NF 11418892 Ki = 3060 nM T94131 CL3Z4O 11419728 Ki = 20 nM T94131 CYBD21 11428504 IC50 = 100000 nM T94131 CHJ30L 11492951 IC50 = 250 nM T94131 C5E2PO 11500850 IC50 = 13500 nM T94131 CV8J3I 11514586 IC50 = 950 nM T94131 CTXF73 11515474 IC50 = 80 nM T94131 C0O4SQ 11522078 IC50 = 30 nM T94131 C7HMO6 11526786 IC50 = 8000 nM T94131 C15XPT 11529859 IC50 = 43 nM T94131 C5KV8L 11530037 IC50 = 530 nM T94131 CGK17J 11536358 IC50 = 110 nM T94131 C38YWS 11541283 IC50 = 6 nM T94131 C1VA4C 11543481 IC50 = 970 nM T94131 C4T8IQ 11550986 IC50 = 290 nM T94131 C63TOQ 11551198 IC50 = 39 nM T94131 CN2MS6 11562853 IC50 = 1258.93 nM T94131 C9JF1G 11565677 IC50 = 2600 nM T94131 CPXS32 11566902 IC50 = 56 nM T94131 CMVQ43 11576772 IC50 = 20 nM T94131 CUZP58 11580302 IC50 = 1000 nM T94131 CX92QM 11581007 IC50 = 29 nM T94131 CEHZ82 11599141 IC50 = 794.33 nM T94131 C6U0BN 11601532 IC50 > 10000 nM T94131 CL5F3Z 11601890 IC50 = 20 nM T94131 C58QVA 11601930 IC50 = 37 nM T94131 C1ZPM5 11630874 IC50 = 30 nM T94131 CLK3Y4 11638999 IC50 = 1000 nM T94131 CU2CK3 11644621 IC50 = 840 nM T94131 CQIX52 11645168 IC50 = 260 nM T94131 C08DUS 11645350 IC50 = 20000 nM T94131 CC64OJ 11652531 IC50 = 40 nM T94131 CP04JC 11666231 IC50 = 2.3 nM T94131 CK8T1S 11666950 IC50 = 29 nM T94131 CU0E8O 11690457 Ki > 4000 nM T94131 CLQ02O 11695207 IC50 = 20000 nM T94131 C3BT1M 11702204 IC50 = 20 nM T94131 CB0AP2 11705863 Ki > 4000 nM T94131 CY8C9P 11751126 IC50 = 382 nM T94131 CAJV97 11955205 IC50 = 21 nM T94131 CBR6D5 11955693 IC50 = 1860 nM T94131 C68SND 11955695 IC50 = 1873 nM T94131 C60DBM 11998444 IC50 > 40000 nM T94131 C5FTB0 11998445 IC50 = 6259 nM T94131 C68WMR 11998447 IC50 = 19790 nM T94131 CYL24B 11998448 IC50 = 16700 nM T94131 CNPI54 11998563 IC50 = 3506 nM T94131 C6AK0Y 11998564 IC50 = 1674 nM T94131 CMVA72 11998565 IC50 = 386 nM T94131 CJ3YP8 11998685 IC50 = 2076 nM T94131 CV8PB5 11998690 IC50 = 829 nM T94131 CB9T1H 11998803 IC50 = 49 nM T94131 C59SKD 11999032 IC50 = 31 nM T94131 CT58GS 12171624 IC50 = 333.96 nM T94131 C0RF3U 14501859 IC50 = 773000 nM T94131 CY7A0T 14638904 IC50 = 10900 nM T94131 CW2XK6 16050925 IC50 = 390 nM T94131 CW5FD8 16081736 IC50 = 16060 nM T94131 C2IF3P 16678352 IC50 > 30000 nM T94131 C3IO1C 16679060 IC50 > 30000 nM T94131 CV9US5 16736978 IC50 > 30000 nM T94131 C72THB 16739368 IC50 = 250 nM T94131 CF6JS9 16757570 IC50 = 54 nM T94131 CB19TH 16757576 IC50 = 10000 nM T94131 C9BJ7Q 16757577 IC50 = 660 nM T94131 C9DM4T 16757578 IC50 = 230 nM T94131 C1NZC7 16757579 IC50 > 10000 nM T94131 CY0S6G 17751063 IC50 = 127 nM T94131 CTP62W 17755300 IC50 = 9000 nM T94131 CQYN41 17755304 IC50 = 3000 nM T94131 C1G7NC 17755392 IC50 = 32700 nM T94131 CI87FV 17755495 IC50 = 17000 nM T94131 CI71OB 17755611 IC50 = 51000 nM T94131 C9W7ID 17755613 IC50 = 12.6 nM T94131 C1SN9M 17756679 IC50 >= 100000 nM T94131 CJAM62 18452190 IC50 = 11.2 nM T94131 C48LCH 18452193 IC50 = 4.27 nM T94131 CVH65S 18452195 IC50 = 2.66 nM T94131 C31KPH 18452198 IC50 = 4.76 nM T94131 CPSJ85 18452200 IC50 = 6.57 nM T94131 C14WMZ 18452237 IC50 = 2.59 nM T94131 CQ89PW 18452323 IC50 = 7.16 nM T94131 C1O3CJ 18452350 IC50 = 23 nM T94131 CXFA80 18452409 IC50 = 37.3 nM T94131 C9Q0EK 18452424 IC50 = 27.5 nM T94131 C5WV4J 18452430 IC50 = 103.4 nM T94131 CVDL81 22036885 IC50 = 6 nM T94131 C61ZGT 22135435 IC50 > 50118.72 nM T94131 CC5QS1 22263527 IC50 = 10890 nM T94131 CP05ZB 22346757 IC50 = 50000 nM T94131 C1F2TM 23582995 IC50 = 1500 nM T94131 CEYL29 23585510 Ki = 88 nM T94131 CR08WX 23586742 IC50 = 7260 nM T94131 CBL37C 23642173 Ki = 1020 nM T94131 C8J1SI 23642272 IC50 = 5285 nM T94131 C59CTR 23652981 IC50 = 97 nM T94131 C29SFI 24768579 IC50 = 829 nM T94131 C3M1OC 24802861 IC50 = 230 nM T94131 CP4G9Z 24855584 Ki = 120 nM T94131 CJV7D9 24855887 IC50 = 50 nM T94131 CM9C0R 24866805 IC50 = 6800 nM T94131 CB79YC 24905143 IC50 = 1500 nM T94131 C2DC9J 24905144 IC50 = 570 nM T94131 CN6V8Z 24905145 IC50 = 100 nM T94131 CSB7P5 24905148 IC50 = 2400 nM T94131 CGSF21 24905149 IC50 = 200 nM T94131 CVDG02 24905150 IC50 = 1800 nM T94131 CWH6C5 24905152 IC50 = 43 nM T94131 C0HE2Q 24905153 IC50 = 72 nM T94131 C7QSC9 24905154 IC50 = 990 nM T94131 CO9D0K 24905155 IC50 = 860 nM T94131 C5W9UR 24905157 IC50 = 1400 nM T94131 CC1DA3 24905158 IC50 = 940 nM T94131 COW79F 24905159 IC50 = 680 nM T94131 CFPA53 24905160 IC50 = 2400 nM T94131 C2O0JX 24905161 IC50 = 7200 nM T94131 CA72BE 24905162 IC50 = 900 nM T94131 CQN6X9 24905163 IC50 = 2400 nM T94131 CD4O1F 24905165 IC50 = 5900 nM T94131 CKL48T 24905166 IC50 = 10000 nM T94131 C76VYL 24905167 IC50 = 1300 nM T94131 C7K5PU 24905168 IC50 = 1400 nM T94131 CZ57ID 24905169 IC50 = 1100 nM T94131 C2DHX9 24905170 IC50 = 2300 nM T94131 CSB96E 24905171 IC50 = 100000 nM T94131 CWZ0R2 24905172 IC50 = 1100 nM T94131 CY3B6M 24905175 IC50 = 551 nM T94131 CW7UA3 24905176 IC50 = 821 nM T94131 CW1V0H 24905177 IC50 = 100000 nM T94131 CO6Y0L 24905178 IC50 = 100000 nM T94131 C60NQW 24905179 IC50 = 8020 nM T94131 C4MO8B 24905180 IC50 = 1470 nM T94131 COJI47 24905181 IC50 = 1210 nM T94131 CS0B2C 24905182 IC50 = 640 nM T94131 C1H4BT 24905183 IC50 = 271 nM T94131 C4WHK9 24905184 IC50 = 4250 nM T94131 C7Q4MZ 24905185 IC50 = 799 nM T94131 CS4IP1 24905186 IC50 = 270 nM T94131 C69QWO 24905187 IC50 = 873 nM T94131 C85ANB 24905188 IC50 = 123 nM T94131 CNHD75 24905189 IC50 = 87 nM T94131 C9JUO2 24905190 IC50 = 1022 nM T94131 CPR03K 24905191 IC50 = 1140 nM T94131 CTAG19 24905193 IC50 = 435 nM T94131 C7VJM5 24905194 IC50 = 430 nM T94131 CEP1L3 24905195 IC50 = 347 nM T94131 CP68ZD 24905196 IC50 = 239 nM T94131 C8Z0RJ 24905197 IC50 = 381 nM T94131 CN9RT0 24905198 IC50 = 100000 nM T94131 CHI78P 24905200 IC50 = 2700 nM T94131 CO6PE8 24905201 IC50 = 2000 nM T94131 CZ63HS 24905202 IC50 = 1300 nM T94131 C2X0FC 24905203 IC50 = 330 nM T94131 C0WCE3 24905204 IC50 = 220 nM T94131 CNK50B 24905205 IC50 = 590 nM T94131 C12DPB 24905206 IC50 = 830 nM T94131 C8N0RH 24905207 IC50 = 2700 nM T94131 CYA5G2 24905208 IC50 = 461 nM T94131 CDV2B4 24905209 IC50 = 1800 nM T94131 CEFK68 24905210 IC50 = 640 nM T94131 CUFP12 24905211 IC50 = 1300 nM T94131 C0JG8L 24905212 IC50 = 1500 nM T94131 CP47MK 24905213 IC50 = 15000 nM T94131 CB61QC 24905214 IC50 = 3000 nM T94131 CQ13ZI 24905215 IC50 = 100000 nM T94131 C6VI8F 24905216 IC50 = 184 nM T94131 CXNH25 24905217 IC50 = 167 nM T94131 C2PN9S 24905218 IC50 = 95 nM T94131 C9O2AL 24905219 IC50 = 228 nM T94131 CIT7U8 24905220 IC50 = 100000 nM T94131 CMD26S 24905221 IC50 = 627 nM T94131 C4R8WC 24905222 IC50 = 31000 nM T94131 C47SHA 24905223 IC50 = 113 nM T94131 C1DY2R 24905224 IC50 = 90 nM T94131 CS0XF9 24905225 IC50 = 100000 nM T94131 CG5VX2 24905226 IC50 = 100000 nM T94131 C57QEO 24905227 IC50 = 100000 nM T94131 C7CG5E 24905228 IC50 = 586 nM T94131 CHP5D1 24905229 IC50 = 3000 nM T94131 CXP09S 24905230 IC50 = 60 nM T94131 CY7XG1 24905231 IC50 = 7300 nM T94131 C7JFQ2 24905232 IC50 = 242 nM T94131 C2JM1P 24905233 IC50 = 6900 nM T94131 CC3BF0 24905234 IC50 = 3000 nM T94131 CE57FI 24905235 IC50 = 4200 nM T94131 CUP20O 24905236 IC50 = 3500 nM T94131 CLC6Q2 24905237 IC50 = 6200 nM T94131 C9M1GI 24905238 IC50 = 2400 nM T94131 CVD72F 24905239 IC50 = 101 nM T94131 CK38IZ 24905240 IC50 = 28 nM T94131 CO2V5E 24905241 IC50 = 22000 nM T94131 CZBA19 24905244 IC50 = 625 nM T94131 CQ8OI1 24905246 IC50 = 100000 nM T94131 C5URC6 24905247 IC50 = 4000 nM T94131 C03SVO 24905250 IC50 = 7700 nM T94131 CIF2J5 24905251 IC50 = 700 nM T94131 CPTE58 24905252 IC50 = 1450 nM T94131 CX1JB8 24905253 IC50 = 2400 nM T94131 COZ3H7 24905254 IC50 = 25000 nM T94131 CDT1H9 24905255 IC50 = 15000 nM T94131 C54QKA 24905256 IC50 = 1700 nM T94131 CRU3P2 24905257 IC50 = 100000 nM T94131 C9U0JA 24905259 IC50 = 11000 nM T94131 CO4YS7 24905260 IC50 = 9600 nM T94131 CEG0B5 24905261 IC50 = 100000 nM T94131 C9VE5F 24905262 IC50 = 100000 nM T94131 C3I4HK 24905264 IC50 = 20000 nM T94131 C0VMI6 24905265 IC50 = 100000 nM T94131 CWE3V0 24905267 IC50 = 100000 nM T94131 CH4T3A 24905268 IC50 = 50000 nM T94131 C6QDN7 24905271 IC50 = 3600 nM T94131 C6XHJ7 24905272 IC50 = 4500 nM T94131 CTB9A3 24905273 IC50 = 17000 nM T94131 C0NB1Q 24905274 IC50 = 6300 nM T94131 C9KQ0L 24905275 IC50 = 5100 nM T94131 C9O8QZ 24905277 IC50 = 4000 nM T94131 CP50RD 24905280 IC50 = 209 nM T94131 CG13ZM 24905281 IC50 = 735 nM T94131 CF0S6X 24905282 IC50 = 5160 nM T94131 C5HBL0 24905284 IC50 = 3340 nM T94131 C2Z5DN 24905285 IC50 = 852 nM T94131 CL6GH8 24905286 IC50 = 523 nM T94131 CKYO98 24905287 IC50 = 435 nM T94131 CRNQ65 24905288 IC50 = 340 nM T94131 COD7I5 24905289 IC50 = 772 nM T94131 C4LP7E 24905290 IC50 = 550 nM T94131 CE9JC2 24905291 IC50 = 200 nM T94131 C2GI1R 24905292 IC50 = 909 nM T94131 CHW8C4 24905293 IC50 = 355 nM T94131 CQF0H1 24905294 IC50 = 120 nM T94131 CNO7X0 24905295 IC50 = 140 nM T94131 C5WRG7 24905296 IC50 = 116 nM T94131 CQ1S0U 24905297 IC50 = 311 nM T94131 C4UES7 24905298 IC50 = 353 nM T94131 CMS69P 24905299 IC50 = 12500 nM T94131 CC0U5M 24905300 IC50 = 147 nM T94131 CW7X6S 24905301 IC50 = 16400 nM T94131 C97IQV 24905302 IC50 = 257 nM T94131 CSJ47V 24905303 IC50 = 1530 nM T94131 CPN74C 24905304 IC50 = 1820 nM T94131 C5CS3N 24905305 IC50 = 1390 nM T94131 CK4XE9 24905307 IC50 = 1070 nM T94131 CTU6Z3 24905308 IC50 = 100000 nM T94131 C9SQX1 24905309 IC50 = 780 nM T94131 CM75JP 24905310 IC50 = 1190 nM T94131 C9Q2BJ 24905311 IC50 = 1270 nM T94131 C9VUA1 24905312 IC50 = 366 nM T94131 CU3RS1 24905313 IC50 = 460 nM T94131 CYG3H2 24905314 IC50 = 633 nM T94131 CV5Q7O 24905315 IC50 = 283 nM T94131 C8SA3O 24905316 IC50 = 113 nM T94131 CI5MN3 24905317 IC50 = 58 nM T94131 CJ1P7K 24905318 IC50 = 43 nM T94131 C1T6YQ 24905319 IC50 = 554 nM T94131 CAU86X 24905320 IC50 = 342 nM T94131 C54ISY 24905321 IC50 = 808 nM T94131 C2GE5I 24905322 IC50 = 637 nM T94131 C8D6YK 24905323 IC50 = 606 nM T94131 C5NZH9 24905324 IC50 = 80 nM T94131 C9D6JR 24905325 IC50 = 1070 nM T94131 CLZT41 24905326 IC50 = 293 nM T94131 CW8FD3 24905327 IC50 = 808 nM T94131 CHB7A2 24905328 IC50 = 502 nM T94131 CA8EI3 24905329 IC50 = 448 nM T94131 CCQ0O7 24905330 IC50 = 1080 nM T94131 CJ81AS 24905331 IC50 = 39 nM T94131 C8PW4H 24905332 IC50 = 44 nM T94131 C2Y5TF 24905333 IC50 = 54 nM T94131 CH9FL5 24905334 IC50 = 2300 nM T94131 C1S0PC 24905335 IC50 = 1900 nM T94131 C8N9MV 24905336 IC50 = 7900 nM T94131 C9E8BJ 24905338 IC50 = 4000 nM T94131 CKZ80E 24905342 IC50 = 340 nM T94131 CO8SH1 24905343 IC50 = 200 nM T94131 C7IZL6 24905344 IC50 = 890 nM T94131 CLD3X6 24936051 IC50 = 47 nM T94131 C43VSW 24936353 IC50 = 501.19 nM T94131 C98MEW 24946175 IC50 = 6.7 nM T94131 CC7H3U 24946706 IC50 = 5.2 nM T94131 C78NJE 24955795 IC50 = 3130 nM T94131 C8P6NT 24956158 IC50 = 854 nM T94131 CJI29P 24956159 IC50 = 6654 nM T94131 C6C4RH 24993871 IC50 = 19 nM T94131 CL0TI6 24993895 IC50 = 6165.95 nM T94131 CS3Q8B 24995659 Ki > 4000 nM T94131 C8W3FZ 25023762 IC50 = 77.7 nM T94131 CZ9WE5 25023763 IC50 = 29.5 nM T94131 C3RL8W 25023764 IC50 = 36.1 nM T94131 CI6M9D 25023765 IC50 = 43.7 nM T94131 CF76VL 25023766 IC50 = 2.79 nM T94131 CC1KV3 25023767 IC50 = 2.34 nM T94131 CX7HP1 25023768 IC50 = 18.4 nM T94131 CEO7L0 25023769 IC50 = 33.2 nM T94131 CPA38V 25023770 IC50 = 1.92 nM T94131 C6QML7 25023771 IC50 = 4.28 nM T94131 C3VI4L 25023772 IC50 = 4.96 nM T94131 C6IOR9 25023773 IC50 = 4.84 nM T94131 CEW91Q 25032963 IC50 = 20 nM T94131 CY50OT 25052783 IC50 = 78 nM T94131 CHR51O 25057242 IC50 = 2600 nM T94131 CTM16Y 25069911 IC50 = 7909 nM T94131 CVI2S5 25070227 IC50 = 7582 nM T94131 CNL4Y2 25070228 IC50 = 11000 nM T94131 CSDN18 25070229 IC50 = 7907 nM T94131 CK92QL 25070230 IC50 = 10322 nM T94131 CKZ7X2 25070231 IC50 = 5830 nM T94131 C0T4NK 25070551 IC50 = 683 nM T94131 C1UKQ4 25070552 IC50 = 1378 nM T94131 CZRA03 25070553 IC50 = 2378 nM T94131 CO20FT 25070554 IC50 = 10000 nM T94131 CL4B5Z 25070555 IC50 = 1650 nM T94131 C7U0SC 25070882 IC50 = 1134 nM T94131 CCN36H 25071204 IC50 = 44 nM T94131 CQ7P4X 25071206 IC50 = 119 nM T94131 C14SFA 25071208 IC50 = 204 nM T94131 CNCJ40 25071516 IC50 = 61 nM T94131 CXWO13 25071518 IC50 = 776 nM T94131 CBH13R 25071519 IC50 = 1102 nM T94131 CJM7O0 25071520 IC50 = 594 nM T94131 C68PFD 25073081 IC50 = 583 nM T94131 CBJ20X 25073385 IC50 = 306 nM T94131 CZN7W0 25073388 IC50 = 368 nM T94131 CD69RK 25097993 IC50 = 33 nM T94131 CLP07J 25110819 IC50 > 10000 nM T94131 CVM89J 25128663 IC50 = 79.43 nM T94131 C4HRL9 25128667 IC50 = 39.81 nM T94131 C4SWT5 25128668 IC50 = 158.49 nM T94131 CIO6A4 25129024 IC50 = 630.96 nM T94131 CLS7P0 25129381 IC50 = 1995.26 nM T94131 C9R2EA 25129383 IC50 = 3981.07 nM T94131 C4YZL9 25129386 IC50 = 316.23 nM T94131 CDO9Q0 25129729 IC50 = 3981.07 nM T94131 CX86YV 25129734 IC50 = 398.11 nM T94131 CA2K4U 25130429 IC50 = 316.23 nM T94131 C1J8KH 25132804 IC50 = 3981.07 nM T94131 CI04XW 25132806 IC50 = 1000 nM T94131 C5WC4L 25133141 IC50 = 251.19 nM T94131 CSH37X 25133142 IC50 = 63.1 nM T94131 CW3HN6 25133144 IC50 = 1584.89 nM T94131 C4LHV1 25165368 IC50 > 10000 nM T94131 C2CXH3 25165371 IC50 > 10000 nM T94131 CQWL59 25165372 IC50 > 10000 nM T94131 CL87JW 25165773 IC50 = 7000 nM T94131 CB89TL 25165774 IC50 > 10000 nM T94131 CFZI92 25165961 IC50 > 10000 nM T94131 CK2YI4 25168990 IC50 = 6309.57 nM T94131 CC1D8V 25172062 IC50 = 14 nM T94131 CPW2D9 25172477 IC50 = 11 nM T94131 CLW96O 25207689 IC50 = 15 nM T94131 CWP29U 25242324 IC50 = 16 nM T94131 C4V2EJ 25261231 IC50 = 148 nM T94131 C3IDN0 25266674 IC50 = 12589.25 nM T94131 CIXE02 28063903 IC50 = 915000 nM T94131 C2IM0O 39733146 IC50 = 2511.89 nM T94131 CO4PL8 42606076 IC50 > 100000 nM T94131 C20VGT 42606077 IC50 = 40000 nM T94131 C7N5EC 42606078 IC50 > 100000 nM T94131 CIF63E 42623219 IC50 = 100 nM T94131 C3DNM9 42623223 IC50 = 25.12 nM T94131 COR5I0 42623224 IC50 = 251.19 nM T94131 CX1DC2 42623385 IC50 = 6.31 nM T94131 CR6N3I 42623632 IC50 = 15.85 nM T94131 C4EM0W 42623869 IC50 = 630.96 nM T94131 C5TY9Q 42623950 IC50 = 158.49 nM T94131 C10RBA 42636535 IC50 = 8000 nM T94131 C8N6CY 44119296 IC50 = 156000 nM T94131 C3ROX1 44124863 Ki = 1.9 nM T94131 CI3K7H 44129042 IC50 = 7900 nM T94131 CIE0J3 44129043 IC50 > 10000 nM T94131 CUW85V 44129044 IC50 > 10000 nM T94131 C2B9DE 44129118 IC50 = 8300 nM T94131 C0R1PH 44129198 IC50 > 10000 nM T94131 C6LGD5 44129200 IC50 = 3000 nM T94131 C03RLS 44129270 IC50 > 10000 nM T94131 CU4H1I 44129274 IC50 > 10000 nM T94131 C79QOC 44129275 IC50 = 6100 nM T94131 C0W3ZF 44129348 IC50 > 10000 nM T94131 CH6RO4 44129351 IC50 > 10000 nM T94131 CPAU59 44129353 IC50 > 10000 nM T94131 CN5O4I 44129429 IC50 = 2900 nM T94131 C3ZSV2 44129432 IC50 = 6300 nM T94131 CM5U2I 44137407 IC50 = 211 nM T94131 CQ82MS 44138035 IC50 = 23000 nM T94131 CZA3N9 44138128 IC50 = 34000 nM T94131 CF17OS 44180029 IC50 = 808 nM T94131 CHK8Z6 44180034 IC50 = 1170 nM T94131 CEJ5F7 44180035 IC50 = 9180 nM T94131 CQNT23 44180155 IC50 = 158 nM T94131 CIKM57 44180156 IC50 = 1310 nM T94131 CBP2T3 44180157 IC50 = 1090 nM T94131 C9CGB4 44180282 IC50 = 503 nM T94131 C2S5LC 44180395 IC50 = 410 nM T94131 C40NOQ 44180397 IC50 = 1080 nM T94131 CTB46H 44180398 IC50 = 547 nM T94131 CRS2G3 44180853 IC50 = 3945 nM T94131 C2VZX7 44181492 IC50 > 50000 nM T94131 C7SYM2 44181493 IC50 = 8780 nM T94131 CB8KF1 44181494 IC50 = 5460 nM T94131 C5AI8R 44181598 IC50 = 4220 nM T94131 CK03RW 44181599 IC50 = 2310 nM T94131 CXL61J 44181600 IC50 = 1570 nM T94131 C6TZK5 44181601 IC50 = 385 nM T94131 CCIV74 44181602 IC50 = 553 nM T94131 C36WUP 44181603 IC50 > 50000 nM T94131 CS2U7R 44181604 IC50 = 6300 nM T94131 CL6W0C 44181605 IC50 = 314 nM T94131 CFD41Z 44181718 IC50 = 7500 nM T94131 C2RB1P 44181719 IC50 = 5200 nM T94131 CMC75I 44181720 IC50 = 1390 nM T94131 CWTS93 44181721 IC50 = 667 nM T94131 CT1JL2 44181722 IC50 = 586 nM T94131 CE9HO1 44181723 IC50 = 5560 nM T94131 CFSB29 44181724 IC50 = 4990 nM T94131 CS0M9A 44187604 IC50 = 18.5 nM T94131 C0BRI9 44187779 IC50 = 37 nM T94131 CDA81B 44187783 IC50 = 25 nM T94131 C0LB8S 44187784 IC50 = 11.5 nM T94131 CCTO21 44187951 IC50 = 84.5 nM T94131 CVYS60 44187952 IC50 = 12 nM T94131 C8X3UZ 44187955 IC50 = 9 nM T94131 CJU85Z 44188321 IC50 = 33 nM T94131 CHU02A 44188322 IC50 = 17.2 nM T94131 C69HQS 44188840 IC50 = 13.5 nM T94131 CD78AG 44188841 IC50 = 19.5 nM T94131 CY7EL1 44188842 IC50 = 21.5 nM T94131 C0SE1X 44188843 IC50 = 48.5 nM T94131 CG13ZF 44188844 IC50 = 24.8 nM T94131 CR0BF9 44189010 IC50 = 78 nM T94131 C71NFL 44189011 IC50 = 69 nM T94131 C39ABJ 44189192 IC50 = 17.5 nM T94131 CK73NR 44219749 IC50 = 6315 nM T94131 CZ3L7W 44233390 IC50 = 1697 nM T94131 CA7R1U 44233391 IC50 = 1772 nM T94131 CU2F9E 44413107 IC50 = 29 nM T94131 C9SK8P 44413114 IC50 = 200 nM T94131 C9ZML1 44454396 IC50 = 117 nM T94131 CVG75D 44473371 IC50 = 8 nM T94131 C30NZA 44475985 IC50 = 69 nM T94131 CAT8F7 44475986 IC50 = 185 nM T94131 CSR73H 44475987 IC50 = 1300 nM T94131 CDAX92 44475988 IC50 = 113 nM T94131 CBH0S5 44475989 IC50 = 20000 nM T94131 CW5A7L 44475990 IC50 = 4 nM T94131 CLKU13 44481151 Ki = 39 nM T94131 CX3FK1 44513884 IC50 = 28.5 nM T94131 CL4RO5 44513885 IC50 = 34 nM T94131 C6RC9J 44513886 IC50 = 27 nM T94131 CGS7Q4 44513887 IC50 = 23 nM T94131 CSVD32 44513888 IC50 = 438 nM T94131 CLN2M5 44514201 IC50 = 52.5 nM T94131 C2Y8ML 44514203 IC50 = 219.5 nM T94131 CA9H8D 44514205 IC50 = 528 nM T94131 C01ZJI 44514208 IC50 = 18 nM T94131 CZ8WK6 44514210 IC50 = 24.5 nM T94131 CI8H3K 44514481 IC50 = 814.5 nM T94131 C51SEJ 44515083 IC50 = 21.5 nM T94131 CXBV98 44515084 IC50 = 14.5 nM T94131 C73HNB 44515696 IC50 = 85 nM T94131 CB7XW5 44516307 IC50 = 48.5 nM T94131 C4W5EM 44516309 IC50 = 9 nM T94131 C8VAU1 44516310 IC50 = 20 nM T94131 C8I1ZB 44516311 IC50 = 9 nM T94131 CSJ95V 44516635 IC50 = 10 nM T94131 CV6Z0N 44516636 IC50 = 10 nM T94131 CB3MV8 44517288 IC50 = 49.5 nM T94131 CDEQ97 44520808 IC50 = 993 nM T94131 CB4RN0 44520812 IC50 = 2367 nM T94131 CFC65B 44539960 IC50 <= 1000 nM T94131 C03IGD 44540030 IC50 = 7943.28 nM T94131 C5LWU1 44540126 IC50 = 7943.28 nM T94131 CYD4Z8 44540130 IC50 = 50.12 nM T94131 CAT2R7 44540316 IC50 = 15848.93 nM T94131 C36NRP 44540403 IC50 <= 1000 nM T94131 C2T9GC 44540407 IC50 = 6309.57 nM T94131 CQ4PE7 44540492 IC50 > 25118.86 nM T94131 C6HC3L 44548482 IC50 = 72.5 nM T94131 CH3L9P 44551660 IC50 > 1000 nM T94131 CYMD49 44552663 IC50 = 1358 nM T94131 C6B7LH 44552664 IC50 = 473 nM T94131 C3QZX0 44552666 IC50 = 283 nM T94131 C64OQC 44552667 IC50 = 155 nM T94131 C7LG6Q 44552844 IC50 = 404 nM T94131 C9T2CZ 44552845 IC50 = 76 nM T94131 CXLD75 44552846 IC50 = 109 nM T94131 CALT95 44554240 IC50 = 2781 nM T94131 CVDA08 44554755 IC50 = 1458 nM T94131 C25EGX 44554909 IC50 = 1820 nM T94131 CR4J0X 44554913 IC50 = 1625 nM T94131 CWV2T9 44554915 IC50 = 402 nM T94131 CCW12H 44555222 IC50 = 269 nM T94131 CTM8S9 44555225 IC50 = 2419 nM T94131 C7PSO6 44555226 IC50 = 646 nM T94131 C3VRO9 44557921 IC50 = 12.59 nM T94131 CRE61W 44577592 IC50 = 258 nM T94131 CH63GM 44577593 IC50 = 113 nM T94131 CA8MV5 44577594 IC50 = 321 nM T94131 C9IXW8 44577638 IC50 = 159 nM T94131 C8A5RT 44577639 IC50 = 28 nM T94131 CNP02V 44577640 IC50 = 73 nM T94131 CT6GN5 44577641 IC50 = 189 nM T94131 CIQR97 44577850 IC50 = 959 nM T94131 CCG8P9 44577851 IC50 = 16840 nM T94131 CLBA40 44577853 IC50 = 357 nM T94131 COU6V7 44577854 IC50 = 531 nM T94131 C8M5FY 44577914 IC50 = 318 nM T94131 C3MGZ9 44577915 IC50 > 20000 nM T94131 CGO09K 44577916 IC50 = 80 nM T94131 CRJ3B7 44577917 IC50 = 210 nM T94131 CTR89C 44577918 IC50 > 20000 nM T94131 CO05YG 44577919 IC50 = 163 nM T94131 CT70WA 44577920 IC50 = 77 nM T94131 C5KXS4 44577921 IC50 = 145 nM T94131 CZ2HI5 44577922 IC50 = 107 nM T94131 CGTU34 44577950 IC50 = 819 nM T94131 CQC50R 44577951 IC50 = 52 nM T94131 C8ZTW2 44577952 IC50 = 440 nM T94131 CIL93G 44577953 IC50 = 617 nM T94131 C8NB5H 44578037 IC50 > 40000 nM T94131 CX9TO2 44578038 IC50 = 35730 nM T94131 C7AHR4 44578039 IC50 > 50000 nM T94131 C13LGI 44578040 IC50 > 50000 nM T94131 CNZ06H 44578074 IC50 > 50000 nM T94131 C41TYA 44578108 IC50 = 63 nM T94131 C2W3SQ 44578109 IC50 = 223 nM T94131 CYM69I 44580064 IC50 = 51 nM T94131 CV09JM 44580065 IC50 = 34 nM T94131 CF37TO 44580066 IC50 = 35 nM T94131 CA0BU6 44580067 IC50 = 203 nM T94131 COQ85J 44580235 IC50 = 24 nM T94131 CD4ER0 44580236 IC50 = 20 nM T94131 CHVQ28 44580237 IC50 = 34 nM T94131 C8N2AF 44580238 IC50 = 767 nM T94131 C40LVX 44580274 IC50 = 1288 nM T94131 CO9LD8 44580275 IC50 = 138 nM T94131 C5QWG4 44580276 IC50 = 222 nM T94131 CFZS45 44580277 IC50 = 174 nM T94131 CQ4CR6 44580635 IC50 = 201 nM T94131 CJHK57 44580636 IC50 = 257 nM T94131 CC6M2E 44580684 IC50 = 70 nM T94131 CA3KP5 44580685 IC50 = 180 nM T94131 C40VHS 44580686 IC50 = 52 nM T94131 CXV92J 44580687 IC50 = 767 nM T94131 CG3PH2 44580721 IC50 = 327 nM T94131 CIO46B 44580722 IC50 = 48 nM T94131 CNLS71 44580723 IC50 = 35 nM T94131 C1N0MF 44580724 IC50 = 18 nM T94131 CAHQ76 44580766 IC50 = 131 nM T94131 C2XN6B 44580767 IC50 = 51 nM T94131 CC36YN 44580768 IC50 = 70 nM T94131 CZ56FY 44580769 IC50 = 46 nM T94131 CL8S0Y 44592136 IC50 >= 50000 nM T94131 C9E6JV 44592170 IC50 = 10000 nM T94131 C8DUA1 44592171 IC50 < 10000 nM T94131 CY8VU1 44592172 IC50 < 10000 nM T94131 C56TOC 44592173 IC50 < 10000 nM T94131 CGP6M7 44592216 IC50 >= 100000 nM T94131 CS38JL 44592217 IC50 = 100000 nM T94131 CJ1FW0 44592218 IC50 > 100000 nM T94131 C70VRG 44592219 IC50 > 100000 nM T94131 CW5RQ0 44592258 IC50 > 100000 nM T94131 CVB1I3 44592259 IC50 > 100000 nM T94131 CV9MY8 44592260 IC50 > 100000 nM T94131 CA65CE 44592261 IC50 > 100000 nM T94131 CEHY48 44592262 IC50 > 100000 nM T94131 C09OLK 44592299 IC50 = 42000 nM T94131 CJM35R 44592300 IC50 > 100000 nM T94131 C54DKW 44592302 IC50 = 42000 nM T94131 CJX76V 44592338 IC50 > 100000 nM T94131 CNY53M 44592339 IC50 > 100000 nM T94131 CXPK04 44592340 IC50 > 100000 nM T94131 C0L2HO 44593630 IC50 = 107 nM T94131 C2NQ6Z 44593631 IC50 = 22 nM T94131 CHKQ45 44593990 IC50 > 10000 nM T94131 CY3SV7 44596118 IC50 > 10000 nM T94131 C28QLM 44605035 IC50 = 6224 nM T94131 C75XHS 44605037 IC50 = 495 nM T94131 C3F4UX 44605249 IC50 = 1431 nM T94131 CQ0FZ7 44605426 IC50 = 3765 nM T94131 CC7G2L 44605427 IC50 = 3554 nM T94131 CDLP04 44605428 IC50 = 409 nM T94131 CSKN09 44605429 IC50 = 2526 nM T94131 CA79QG 44605430 IC50 = 1290 nM T94131 CH6V9F 44608754 IC50 = 6.5 nM T94131 C0IY9N 44608757 IC50 = 16 nM T94131 C90ITS 44608915 IC50 = 8.1 nM T94131 CZH1P9 44609387 IC50 = 2.4 nM T94131 CNDX48 44609388 IC50 = 13 nM T94131 CE95RQ 44620964 IC50 = 15 nM T94131 CVYJ36 44620965 IC50 = 33 nM T94131 CA8BY7 44621440 IC50 = 31.62 nM T94131 C5M1FR 44621441 IC50 = 25.12 nM T94131 C5LD7E 44621442 IC50 = 7.943 nM T94131 CO4GT0 44621447 IC50 = 25.12 nM T94131 CUV26H 44621448 IC50 = 19.95 nM T94131 CV2MG9 44621449 IC50 = 19.95 nM T94131 C24IYW 44621451 IC50 = 39.81 nM T94131 C0F9YW 44621452 IC50 = 100 nM T94131 C0GRD8 44621454 IC50 = 79.43 nM T94131 C4YHJ0 44621456 IC50 = 19.95 nM T94131 C31VBF 44621458 IC50 = 15.85 nM T94131 CQD03G 44623048 Ki = 770 nM T94131 C54IUP 44818842 IC50 = 435 nM T94131 C16IMZ 44819024 IC50 = 49 nM T94131 CN38JF 44819199 IC50 = 48.5 nM T94131 CVW6L8 44819200 IC50 = 22 nM T94131 CZ7M6D 44819201 IC50 = 12.2 nM T94131 C7MU8J 44819203 IC50 = 12.3 nM T94131 C8FU0W 44819375 IC50 = 22 nM T94131 C4N8CK 44819376 IC50 = 25 nM T94131 CP6DB9 45265864 IC50 = 40 nM T94131 C5I1VH 45379222 IC50 = 789 nM T94131 CA4JZ8 45379223 IC50 = 65 nM T94131 CZ68MG 45488079 IC50 > 10000 nM T94131 CV1U7I 46180604 IC50 = 8.4 nM T94131 CED2B3 46180606 IC50 = 5100 nM T94131 CDV85O 46180663 IC50 = 1300 nM T94131 CZGB46 46180666 IC50 = 15 nM T94131 C61ZLI 46190736 IC50 = 265 nM T94131 C6H3GT 46196486 IC50 = 33 nM T94131 CAU17V 46202808 IC50 = 3.162 nM T94131 CDA3R9 46220225 IC50 = 8 nM T94131 CIJ5V9 46224766 IC50 = 223 nM T94131 CIPV59 46224808 IC50 = 640 nM T94131 CRQ5M4 46225259 IC50 = 10000 nM T94131 C65IPQ 46225280 IC50 = 133 nM T94131 C8A7QJ 46225281 IC50 = 341 nM T94131 CPL45H 46225307 IC50 = 6907 nM T94131 CTN8J2 46225308 IC50 = 8297 nM T94131 CL34IK 46227801 IC50 = 510 nM T94131 C6D2RL 46227820 IC50 = 975 nM T94131 CSIK15 46228569 IC50 = 7470 nM T94131 C94YRI 46853654 IC50 = 3.981 nM T94131 CZ3WS1 46861592 IC50 = 5 nM T94131 CRO8W0 46865423 IC50 = 25 nM T94131 C47VTS 46865424 IC50 = 11 nM T94131 CO3P0J 46866604 IC50 = 1256 nM T94131 CQ2Y1V 46866705 Ki = 0.111 nM T94131 C63RCG 46870269 IC50 = 2.512 nM T94131 CTQ25M 46871497 IC50 = 6.31 nM T94131 CXRI03 46872177 Ki = 0.048 nM T94131 CC0R5U 46872178 Ki = 0.017 nM T94131 C8SRB0 46872297 Ki = 0.157 nM T94131 C67QZY 46872298 Ki = 0.33 nM T94131 CQB16A 46872415 Ki = 0.003 nM T94131 C7V8RJ 46873664 Ki = 0.066 nM T94131 CJB8T7 46873665 Ki = 0.011 nM T94131 CU7Z9M 46873667 Ki = 0.013 nM T94131 C6MZ1J 46884121 IC50 = 6949 nM T94131 CLA40T 46885426 IC50 = 3628 nM T94131 CC8T1E 46885496 IC50 = 2220 nM T94131 CCS20H 46885565 IC50 = 10 nM T94131 CG47YP 46885566 IC50 = 587 nM T94131 C4R3XP 46885599 IC50 = 54 nM T94131 CV5MK6 46885601 IC50 = 976 nM T94131 C42WVO 46885648 IC50 = 322 nM T94131 C3HMQ2 46891474 IC50 = 2.4 nM T94131 CB6Z8P 46892208 IC50 = 6200 nM T94131 CZX46Y 46892342 IC50 = 110 nM T94131 C5FN6I 46892845 IC50 = 320 nM T94131 CQ32BN 46892970 IC50 = 8 nM T94131 COJA32 46892971 Ki = 69 nM T94131 C5QFB3 46893088 IC50 = 200 nM T94131 CS30AI 46893754 IC50 = 3600 nM T94131 CPO1N7 46927938 Ki = 179 nM T94131 CJ0VB4 46932297 IC50 = 430 nM T94131 CL84AF 46946248 Ki > 500 nM T94131 CF14PE 46947264 IC50 = 74 nM T94131 COE37N 49778924 IC50 = 790 nM T94131 C7ZK3D 49783923 IC50 = 316.23 nM T94131 CHX76J 49784892 Ki = 29 nM T94131 CA1H8S 49784893 Ki = 88 nM T94131 CP2QD0 49784894 Ki = 4 nM T94131 CTZG05 49784988 Ki = 45 nM T94131 CE9AC5 49785078 Ki = 23 nM T94131 CG2IO7 49785079 Ki = 12 nM T94131 C8EYN4 49785083 Ki = 17 nM T94131 CBNZ47 49785166 Ki = 136 nM T94131 CZI34V 49785167 Ki = 330 nM T94131 CJK65T 49785253 Ki = 51 nM T94131 CXK8F5 49785436 Ki = 2 nM T94131 CWL5C6 49785518 Ki = 6 nM T94131 C3NV0J 49785827 Ki = 12 nM T94131 C0OZM2 49785828 Ki = 200 nM T94131 C1AR4G 49785829 Ki = 450 nM T94131 C39HAK 49785832 Ki = 12 nM T94131 C90JBE 49834576 IC50 > 10000 nM T94131 C5UR4A 49843944 IC50 = 720 nM T94131 CS40YB 49853846 IC50 = 230 nM T94131 C7PER0 49853953 IC50 = 660 nM T94131 CU9A8O 49854022 IC50 > 10000 nM T94131 C51QVH 49854023 IC50 = 10000 nM T94131 CM4HQ2 49854024 IC50 > 10000 nM T94131 C1LBX3 49854049 IC50 = 430 nM T94131 CVC2H6 49854052 IC50 = 290 nM T94131 CC2X9N 49854121 IC50 > 10000 nM T94131 CAJ58E 49854156 IC50 = 180 nM T94131 CAU39Y 49854158 IC50 = 200 nM T94131 CPK6X3 49854360 IC50 = 1400 nM T94131 CBVT70 49854361 IC50 = 4000 nM T94131 CQ1TZ6 49854365 IC50 = 1100 nM T94131 CJ5I9X 49854461 IC50 = 330 nM T94131 CDXQ69 49854462 IC50 = 8000 nM T94131 C0ORZ9 49854466 IC50 = 200 nM T94131 CY14XF 49854572 IC50 = 1200 nM T94131 CEC10T 49854573 IC50 = 15 nM T94131 C39KQW 49854679 IC50 = 200 nM T94131 C8VDR2 49854680 IC50 = 160 nM T94131 CN2V8R 49854681 IC50 = 990 nM T94131 CSN96A 49855001 IC50 = 230 nM T94131 CALY90 49855192 IC50 = 5000 nM T94131 CJPE20 49855193 IC50 = 2500 nM T94131 C1OM3I 49855237 IC50 = 17780 nM T94131 C26IQK 49857091 IC50 = 5300 nM T94131 CR0PN9 49857092 IC50 = 5700 nM T94131 CCJN26 49857093 IC50 = 1900 nM T94131 C3YG5L 49857275 IC50 > 10000 nM T94131 CHO65B 49857279 IC50 = 2640 nM T94131 C9HMY1 49857280 IC50 = 1800 nM T94131 CGW9L1 49857476 IC50 = 5150 nM T94131 CRD84P 49857479 IC50 = 1400 nM T94131 COF78C 49857678 IC50 > 10000 nM T94131 C4H7XG 49857865 IC50 = 2200 nM T94131 CY8MP7 49867926 IC50 = 9 nM T94131 CR0IA5 49871864 IC50 = 1100 nM T94131 C13WJZ 49872243 IC50 = 290 nM T94131 C5OY7B 49872246 IC50 = 146 nM T94131 C2KD5E 49872344 IC50 = 62 nM T94131 CV5BF3 49872645 IC50 = 634 nM T94131 CN97FO 49872646 IC50 = 22.5 nM T94131 CD6P5R 49872735 IC50 = 507 nM T94131 CL64NB 49872737 IC50 = 4650 nM T94131 CRNG04 49872831 IC50 = 11 nM T94131 CQC8B4 49872835 IC50 = 13 nM T94131 CPS3O1 49872924 IC50 = 120 nM T94131 CUBX74 49872925 IC50 = 19 nM T94131 CAW69U 49872927 IC50 = 220 nM T94131 CV1L4P 49873242 IC50 = 964 nM T94131 C5BA2V 49873243 IC50 = 3590 nM T94131 CSN45W 49873329 IC50 = 35.4 nM T94131 CLC2N7 50913517 IC50 = 20500 nM T94131 CJ4L8Y 50938829 Ki = 364 nM T94131 CJG65L 50939078 Ki = 509 nM T94131 CI8QM1 50939080 Ki = 28 nM T94131 CT0IP3 50939081 Ki = 90 nM T94131 C54EUL 50939212 Ki = 7340 nM T94131 CS7Z6U 50939338 Ki = 92 nM T94131 C2I9PS 50939992 IC50 = 18000 nM T94131 C9TUE4 50940108 IC50 = 1400 nM T94131 C2Q0GE 50990922 IC50 = 100 nM T94131 CKY3V1 50990924 Ki = 4.7 nM T94131 C5ZF9W 51003380 IC50 = 77000 nM T94131 CY36EH 51003592 IC50 = 398.11 nM T94131 CLB85F 51346892 IC50 = 740 nM T94131 C65ILG 51346893 IC50 = 44 nM T94131 CRJ5W8 51358113 IC50 = 5.67 nM T94131 CT91WR 52040626 IC50 = 371 nM T94131 CG7T4H 52913198 IC50 = 25 nM T94131 CD84MT 52913592 IC50 = 2200 nM T94131 C2TLG6 52913931 IC50 = 1800 nM T94131 CQ5GF2 52917084 Ki = 126 nM T94131 CAFR91 52917382 Ki = 361 nM T94131 C2DQK4 52917534 Ki = 50.1 nM T94131 C5ON6F 52919356 IC50 = 14 nM T94131 CM5BX0 52919492 IC50 = 68 nM T94131 CU1P2L 52940797 IC50 = 2010 nM T94131 CD62QJ 52940982 IC50 = 358 nM T94131 C43SVQ 52941322 IC50 = 189.5 nM T94131 CK59HM 52941479 IC50 = 150 nM T94131 C2KI6V 52942202 IC50 = 100000 nM T94131 CFRN73 52942850 IC50 = 122 nM T94131 C4D1KT 52942879 IC50 = 44 nM T94131 C4VCY0 52943258 IC50 = 16000 nM T94131 C1XEV2 52943394 IC50 = 2410 nM T94131 C73WTL 52943744 IC50 = 45.2 nM T94131 C6Q1AH 52943745 IC50 = 100 nM T94131 CHI0P6 52944356 IC50 = 100000 nM T94131 CWD27C 52945142 IC50 = 240 nM T94131 CWPC54 52945348 IC50 = 140 nM T94131 CXL53B 52945589 IC50 = 154 nM T94131 C4NLX7 52945630 IC50 = 723 nM T94131 CXD6T8 52945845 IC50 = 1200 nM T94131 CN8F0V 52946289 IC50 = 717 nM T94131 CMQY93 52946368 IC50 = 149 nM T94131 C5X9VO 52948007 IC50 = 290 nM T94131 C7ET6Z 52948010 IC50 = 1600 nM T94131 CW9Z1T 52949347 IC50 = 51 nM T94131 CV5B2C 52949497 IC50 = 25000 nM T94131 CB0KM5 52949869 IC50 = 98 nM T94131 CAJQ03 52950001 IC50 = 99 nM T94131 C5HQ2E 52950102 IC50 = 74 nM T94131 CH1Q5D 53234281 IC50 = 3 nM T94131 C45JKN 53234283 IC50 = 8.4 nM T94131 CVK28S 53235062 IC50 = 0.7 nM T94131 COW61E 53235216 IC50 = 1.5 nM T94131 CWE56X 53235217 IC50 = 3.7 nM T94131 CDXM59 53235451 IC50 = 55 nM T94131 CT8IN1 53242225 IC50 = 3200 nM T94131 C9NF0C 53302364 Ki = 42.4 nM T94131 C4J9WZ 53307606 IC50 = 5 nM T94131 C7ZH0D 53308041 IC50 = 1170 nM T94131 CRD3A9 53316967 IC50 = 340 nM T94131 C84YNK 53317325 IC50 > 83300 nM T94131 CS8DJ3 53318252 IC50 = 150 nM T94131 C58NQJ 53318614 IC50 = 55400 nM T94131 C10YUH 53318615 IC50 = 9700 nM T94131 C24GBF 53319075 IC50 = 15 nM T94131 CFJD70 53319932 IC50 = 70000 nM T94131 C3EJB1 53319933 IC50 = 9100 nM T94131 C2V7AX 53320017 IC50 = 380 nM T94131 CKGJ60 53320018 IC50 = 730 nM T94131 CJRM64 53322563 IC50 = 43500 nM T94131 CN92LK 53322732 IC50 = 9 nM T94131 CJZ29M 53325374 IC50 = 830 nM T94131 C1TE8J 53325515 IC50 = 7600 nM T94131 C6LAI9 53326166 IC50 = 960 nM T94131 CCU75P 53327266 Ki = 6 nM T94131 C1TWE6 53327269 Ki = 3 nM T94131 COSB47 53327579 Ki = 20 nM T94131 C62JOP 53327629 Ki = 4 nM T94131 CCX7M5 53353847 Ki = 20.7 nM T94131 C23HAU 53361718 IC50 = 7.7 nM T94131 CM60WQ 53361719 IC50 = 13 nM T94131 CL69DK 53377727 IC50 = 81 nM T94131 C6Q8RC 53378051 IC50 = 1584.89 nM T94131 CG3C1J 53379513 IC50 = 4.8 nM T94131 CSV9X2 54579940 IC50 = 13 nM T94131 CN51TL 54579941 IC50 = 4100 nM T94131 C7VZU2 54579942 IC50 = 2300 nM T94131 C4R9JB 54579943 IC50 = 610 nM T94131 CG26HQ 54579944 IC50 = 3700 nM T94131 CC5R3O 54580924 IC50 = 340 nM T94131 C3OIY4 54580925 IC50 = 250 nM T94131 C60TYL 54581049 IC50 = 470 nM T94131 CF2UH5 54581983 IC50 = 20 nM T94131 C23EVN 54582916 IC50 = 26 nM T94131 CT2SV7 54583916 IC50 = 480 nM T94131 CY87EC 54583917 IC50 = 30 nM T94131 C8CPI4 54584859 IC50 = 860 nM T94131 C9TZ2V 54584860 IC50 = 2300 nM T94131 CME81Q 54585830 IC50 = 190 nM T94131 CFI7E6 54754350 IC50 = 760 nM T94131 CE4TS9 56589559 IC50 = 32 nM T94131 CR24WQ 56595421 IC50 = 56 nM T94131 CJ41GT 56595686 IC50 = 52 nM T94131 C2PN4S 56599298 IC50 = 6600 nM T94131 CT64SR 56599306 IC50 = 23 nM T94131 CFUT05 56648675 IC50 = 17 nM T94131 C1GAB6 56648677 IC50 = 37 nM T94131 CWDF40 56648757 IC50 = 20 nM T94131 CE35CB 56648758 IC50 = 10 nM T94131 CJO39U 56648759 IC50 = 25 nM T94131 CNKC90 56654649 IC50 > 9100 nM T94131 C83QGP 56660108 IC50 = 9.5 nM T94131 CYM1D0 56660109 IC50 = 6 nM T94131 CHA35L 56663573 IC50 = 4 nM T94131 CF7PY5 56667023 IC50 = 7 nM T94131 CC1DJ8 56670464 IC50 = 20.5 nM T94131 CZH95G 56673952 IC50 = 8 nM T94131 CHR8K0 56677282 IC50 = 10.5 nM T94131 C79AMB 56677283 IC50 = 13.5 nM T94131 CG17TZ 56683916 IC50 = 9.5 nM T94131 C7B2OH 56683917 IC50 = 6.5 nM T94131 C6LMP8 56683918 IC50 = 14.3 nM T94131 C94JIT 56832510 Ki = 0.55 nM T94131 C0IJP8 56927258 IC50 > 6309.57 nM T94131 CM28GU 56928390 IC50 = 280 nM T94131 C9MJG4 56929824 IC50 = 50 nM T94131 CYFB96 56932203 IC50 = 63.1 nM T94131 CJ9R2C 56932209 IC50 = 630.96 nM T94131 C8C2FG 56932238 IC50 = 125.89 nM T94131 CX6Q2K 56932240 IC50 = 10 nM T94131 CPGC81 56947516 Ki = 1 nM T94131 CO6K5Q 56955953 IC50 = 441 nM T94131 CAK91L 56955954 IC50 = 18 nM T94131 C8B6JG 56955955 IC50 = 18 nM T94131 CX4W6G 57325497 IC50 = 1750 nM T94131 CVK5A3 57328247 Ki > 500 nM T94131 CW8B4D 57330208 IC50 = 850 nM T94131 C6JMN9 57345685 IC50 = 1600 nM T94131 CZ7RE0 57345686 IC50 = 1000 nM T94131 CA53SC 57351276 Ki = 183 nM T94131 C9RB7K 57391333 Ki > 500 nM T94131 CH37SE 57391335 Ki > 500 nM T94131 C1GVK3 57391362 IC50 > 4000 nM T94131 C0PR9J 57391364 IC50 > 6300 nM T94131 C6L9HO 57391365 IC50 = 3200 nM T94131 C2QX0T 57391366 IC50 = 1600 nM T94131 CLQ9J1 57391367 IC50 = 1300 nM T94131 CQ1W0C 57393124 IC50 = 7900 nM T94131 CZ0RW2 57393125 IC50 = 1600 nM T94131 COT0L2 57394595 IC50 = 19000 nM T94131 CA93ZE 57394864 IC50 = 3200 nM T94131 C6CL4F 57395172 IC50 = 980 nM T94131 CS14ZH 57396608 Ki > 500 nM T94131 CDG2F3 57396625 IC50 = 3200 nM T94131 CD73TE 57396626 IC50 > 6300 nM T94131 CQRU75 57396627 IC50 > 6300 nM T94131 CI34XH 57396628 IC50 > 6300 nM T94131 CYM02V 57397667 IC50 = 2060 nM T94131 CQO74C 57398382 Ki > 500 nM T94131 CV2Z0C 57398383 Ki > 500 nM T94131 C3Q2ZP 57398390 IC50 > 6300 nM T94131 C56TEZ 57398391 IC50 = 5000 nM T94131 CP9Q4U 57398392 IC50 = 10000 nM T94131 C0O5KE 57398393 IC50 = 320 nM T94131 C3G9HW 57399126 IC50 > 10000 nM T94131 CYE09F 57400062 IC50 = 4000 nM T94131 CN5PY7 57400063 IC50 > 7900 nM T94131 CT0Y7E 57400064 IC50 = 2500 nM T94131 C3Q2NF 57401565 IC50 = 395000 nM T94131 CRO5Z6 57401846 Ki > 500 nM T94131 CM63CS 57401865 IC50 = 1300 nM T94131 CG6M4H 57401867 IC50 > 6300 nM T94131 CP8FY5 57401868 IC50 = 1600 nM T94131 CQ5P4X 57401869 IC50 = 2500 nM T94131 CPG6N5 57402167 IC50 = 1310 nM T94131 C8LKZ3 57402168 IC50 = 1980 nM T94131 CF68RN 57403576 IC50 = 6300 nM T94131 CL2R7T 57403577 IC50 > 6300 nM T94131 CC5N9R 57403578 IC50 > 10000 nM T94131 CZ8M5F 57403579 IC50 = 1600 nM T94131 C5NT7R 57403580 IC50 = 1300 nM T94131 CHBV63 57403581 IC50 = 400 nM T94131 CAC72X 57403582 IC50 > 6300 nM T94131 CQ5Z4S 57404801 IC50 = 39.81 nM T94131 C78YHO 57404804 IC50 = 50.12 nM T94131 CNR95F 57404840 IC50 = 1900 nM T94131 CQ4E8N 57405149 IC50 = 50.12 nM T94131 CA8BT7 57405314 IC50 = 794.33 nM T94131 CI40MW 57405315 IC50 = 501.19 nM T94131 CGN72O 57405485 IC50 = 6.31 nM T94131 C5B9XS 57406164 IC50 = 3.981 nM T94131 CEI2S9 57406702 IC50 = 3162.28 nM T94131 CED47A 57410062 IC50 > 10000 nM T94131 C1BVX6 57411134 IC50 > 10000 nM T94131 C39JSW 57411135 IC50 > 10000 nM T94131 CL8F6Q 57411137 IC50 > 10000 nM T94131 CW97FT 57411139 IC50 > 10000 nM T94131 CU0R3A 57411250 IC50 > 10000 nM T94131 C6C5TU 57411252 IC50 > 10000 nM T94131 CD0W2I 57411254 IC50 = 8135 nM T94131 CW1DA3 57411255 IC50 > 10000 nM T94131 C6U4LO 57411256 IC50 > 10000 nM T94131 CP9G7L 57411366 IC50 = 4203 nM T94131 CC5DO3 57411369 IC50 > 10000 nM T94131 C56RBS 57411372 IC50 > 10000 nM T94131 CX9O3T 57411485 IC50 > 10000 nM T94131 CQBM65 57411486 IC50 > 10000 nM T94131 CK5QX7 57411488 IC50 > 10000 nM T94131 C90LNK 57411715 IC50 > 10000 nM T94131 CPXE40 57411716 IC50 > 10000 nM T94131 CE6RY5 57411836 IC50 > 10000 nM T94131 C5JOX3 57411837 IC50 > 10000 nM T94131 C0I5JM 57419280 IC50 > 10000 nM T94131 CT6XL0 57466811 Ki = 36 nM T94131 CRB5P2 57495287 IC50 > 9100 nM T94131 C59YAC 57495353 IC50 = 2230 nM T94131 CJE19S 57523686 IC50 > 10000 nM T94131 CHIU94 57545876 IC50 = 2.512 nM T94131 C0JQ8P 57584929 Ki = 36 nM T94131 CQU8A1 57585145 Ki = 36 nM T94131 C6L4FZ 57599744 IC50 = 810 nM T94131 CV9J7D 57748162 IC50 = 320 nM T94131 CL57CP 57789333 IC50 = 870 nM T94131 CZ21KP 57900314 IC50 = 2.2 nM T94131 CO20YT 58203712 IC50 = 0.6 nM T94131 C7X0OJ 58203779 IC50 = 8.4 nM T94131 CW1M9X 58203976 IC50 = 36 nM T94131 COFN62 58203995 IC50 = 80 nM T94131 C16GRS 58204034 IC50 = 19.1 nM T94131 CM62NB 58204076 IC50 = 3.5 nM T94131 CGA01N 58204242 IC50 = 4.3 nM T94131 CVR9Q2 58233988 IC50 = 25.12 nM T94131 CB9AH8 58234990 IC50 = 6000 nM T94131 CJ8YI2 58234995 IC50 = 830 nM T94131 CZF3U5 58235016 IC50 = 1000 nM T94131 CM0ND7 58235018 IC50 = 930 nM T94131 C25RXY 58235020 IC50 = 1600 nM T94131 CAY94U 58235030 IC50 = 4200 nM T94131 CAJC03 58235033 IC50 = 710 nM T94131 CN7MZ8 58235039 IC50 = 2600 nM T94131 CPW84H 58235041 IC50 = 630 nM T94131 C70CRN 58235043 IC50 = 3500 nM T94131 C5SQV3 58235052 IC50 = 700 nM T94131 CEZ4T5 58235053 IC50 = 2400 nM T94131 C82LIS 58235061 IC50 = 520 nM T94131 C3SO4E 58235062 IC50 = 530 nM T94131 CZ0SD5 58235073 IC50 = 1200 nM T94131 CQP25T 58235077 IC50 = 700 nM T94131 C0LDZ2 58235079 IC50 = 13000 nM T94131 C2YG5L 58235088 IC50 = 2600 nM T94131 CTVF29 58290044 Ki = 13 nM T94131 CJ6R8Q 59251679 IC50 = 8.2 nM T94131 CWF9Z7 59251848 Ki = 13 nM T94131 CRZ5B1 59251991 IC50 = 1190 nM T94131 C6A3KL 59293676 IC50 = 690 nM T94131 CC14ZL 59293709 IC50 = 1100 nM T94131 C0R3TX 59293715 IC50 = 1400 nM T94131 C9TVC6 59293721 IC50 = 1400 nM T94131 CZ5OV1 59293740 IC50 = 410 nM T94131 CB2Z4R 59293755 IC50 = 830 nM T94131 C8AL6C 59293763 IC50 = 610 nM T94131 CT3CF1 59477024 IC50 = 100 nM T94131 CF6YB8 59477038 IC50 = 3162.28 nM T94131 CK3H9O 59477041 IC50 = 199.53 nM T94131 C7KG5E 59477042 IC50 = 1000 nM T94131 C01DZW 59477048 IC50 = 251.19 nM T94131 CPE9X3 59507470 IC50 = 142 nM T94131 C2X8TY 59548177 Ki = 80 nM T94131 C71GBC 59548184 Ki = 7 nM T94131 CGRO45 59548196 Ki = 210 nM T94131 CD39AG 59548207 Ki = 750 nM T94131 C6KP4G 59548220 Ki = 110 nM T94131 CL82RM 59548221 Ki = 7 nM T94131 CTNU85 59548226 Ki = 54 nM T94131 CLB6N4 59548232 Ki = 1100 nM T94131 C2KBG8 59548236 Ki = 9 nM T94131 CSWV07 59548243 Ki = 130 nM T94131 CN48VL 59548245 Ki = 9 nM T94131 CMT2R0 59548250 Ki = 690 nM T94131 C3I8NE 59548256 Ki = 100 nM T94131 C8W5HT 59548263 Ki = 380 nM T94131 CT8Q5B 59548274 Ki = 8 nM T94131 CBG52T 59548278 Ki = 9 nM T94131 CVF1B2 59548283 Ki = 59 nM T94131 CY31EA 59548284 Ki = 99 nM T94131 CO4GT7 59548288 Ki = 1 nM T94131 CFR7S8 59548302 Ki = 24 nM T94131 CRE8B3 59548316 Ki = 16 nM T94131 CRM20Z 59548320 Ki = 140 nM T94131 CX1KJ9 59548322 Ki = 8 nM T94131 CJE5I4 59548341 Ki = 22 nM T94131 C8O1VS 59548349 Ki = 5 nM T94131 CE9W0K 59548355 Ki = 24 nM T94131 CWC65A 59548356 Ki = 9 nM T94131 CMKP95 59548371 Ki = 9 nM T94131 CC8UV3 59548383 Ki = 12 nM T94131 C4SN3U 59548390 Ki = 21 nM T94131 CD4ET2 59548402 Ki = 58 nM T94131 CES59T 59548403 Ki = 90 nM T94131 CE8P3G 59548407 Ki = 14 nM T94131 CO4K2W 59548419 Ki = 2.2 nM T94131 CSDB78 59548424 Ki = 8 nM T94131 C81FCQ 59548431 Ki = 9 nM T94131 CLGY34 59548453 Ki = 11 nM T94131 CBT21W 59548454 Ki = 91 nM T94131 C9DIB3 59548458 Ki = 9 nM T94131 CJT68K 59548460 Ki = 40 nM T94131 C9LFT3 59548462 Ki = 7 nM T94131 CA47YQ 59548474 Ki = 12 nM T94131 CX8C2U 59548480 Ki = 3600 nM T94131 C8S0ED 59605870 IC50 = 540 nM T94131 C4Y3GL 59609976 IC50 = 441 nM T94131 C1PC0J 59634638 IC50 = 210 nM T94131 CP2UY3 59634686 IC50 = 3530 nM T94131 C1TH2N 59634692 IC50 = 1420 nM T94131 CPA0L2 59634709 IC50 = 5360 nM T94131 C7DC6R 59662371 IC50 = 2398.83 nM T94131 C5S0FG 59662506 IC50 = 5754.4 nM T94131 CBI0M6 59688563 IC50 = 398.11 nM T94131 CUYB59 60148924 IC50 = 6600 nM T94131 CM8PD7 60150509 IC50 = 160 nM T94131 C5KD3Z 60154714 Ki > 10000 nM T94131 CS0L4D 60154996 Ki > 10000 nM T94131 C1UI3P 60155086 Ki = 2600 nM T94131 CX08ON 60155087 Ki = 480 nM T94131 CX8J1I 60155265 Ki = 9 nM T94131 CAT40I 60155266 Ki = 4 nM T94131 CD56VA 60155268 Ki = 21 nM T94131 CCQB56 60155375 IC50 = 10 nM T94131 CH5X2S 60155376 IC50 = 18 nM T94131 C74FEN 60155377 IC50 = 326 nM T94131 CZ6G4B 60155378 IC50 = 39 nM T94131 C10AHQ 60155379 IC50 = 17 nM T94131 C5FI4P 60155451 Ki = 18 nM T94131 CX9G4U 60155452 Ki = 8 nM T94131 C9Q7DE 60155469 IC50 = 26 nM T94131 CH8UY5 60155470 IC50 = 65 nM T94131 C3EDY4 60155471 IC50 = 507 nM T94131 CE0ZX1 60155472 IC50 = 152 nM T94131 CG90MC 60155473 IC50 = 53 nM T94131 C82PVI 60155474 IC50 = 167 nM T94131 CX49FT 60155475 IC50 = 161 nM T94131 CR7EG9 60155538 Ki = 46 nM T94131 CU6YB9 60155539 Ki = 30 nM T94131 CW6N1S 60155552 IC50 = 11 nM T94131 CIB08V 60155553 IC50 = 48 nM T94131 CZE28G 60155554 IC50 = 43 nM T94131 CZD2W7 60155555 IC50 = 31 nM T94131 CO6IU3 60155556 IC50 = 49 nM T94131 C6HN5O 60155557 IC50 = 18 nM T94131 CMQ9G1 60155638 IC50 = 507 nM T94131 CG56KT 60155639 IC50 = 26 nM T94131 CBJ65P 60155640 IC50 = 42 nM T94131 C8OJK0 60155641 IC50 = 5 nM T94131 CT9XJ6 60155642 IC50 = 21 nM T94131 C5BYQ3 60155643 IC50 = 8 nM T94131 C57RBF 60155722 IC50 = 587 nM T94131 CU7J6L 60155723 IC50 = 102 nM T94131 CSZA16 60155724 IC50 = 34 nM T94131 C21DWT 60155725 IC50 = 497 nM T94131 C12CQU 60155726 IC50 = 60 nM T94131 CA5TM3 60155805 IC50 = 20 nM T94131 C60RIO 60155806 IC50 = 6 nM T94131 CIRO73 66493714 IC50 = 167 nM T94131 C71LPV 66493729 IC50 = 302 nM T94131 C54NOW 66552297 IC50 > 100000 nM T94131 CX4HW1 66552298 IC50 > 50118.72 nM T94131 CEJ54A 66552343 IC50 = 501.19 nM T94131 CUQ5Y2 66552345 IC50 > 3981.07 nM T94131 C5F8ZE 66552346 IC50 > 100000 nM T94131 CHQC56 66552347 IC50 = 3162.28 nM T94131 CS6BQ0 66552348 IC50 > 12589.25 nM T94131 CGT2V9 66552407 IC50 = 3981.07 nM T94131 CIJ3C5 66552408 IC50 = 39.81 nM T94131 C6ZFI1 66552410 IC50 > 31622.78 nM T94131 C8S7CM 66552411 IC50 = 316.23 nM T94131 C9A7IK 66552412 IC50 > 39810.72 nM T94131 CRC24S 66552467 IC50 > 100000 nM T94131 CHU5V3 66552468 IC50 > 100000 nM T94131 C46POH 66552523 IC50 = 1995.26 nM T94131 C68LXT 66552524 IC50 = 25118.86 nM T94131 C91JZL 66553214 IC50 = 8280 nM T94131 CUC7B3 66557964 IC50 = 190 nM T94131 C9X2TB 66558056 IC50 = 340 nM T94131 CWZ54O 66600540 Ki = 20 nM T94131 C6Q0KU 66612050 Ki = 34 nM T94131 C1R3SI 66653673 IC50 = 3290 nM T94131 CF8BZ7 66677439 IC50 = 1060 nM T94131 C8L9DK 66743362 Ki = 14 nM T94131 C1IKT2 66743443 Ki = 11 nM T94131 CN0RE8 66779813 IC50 = 1000 nM T94131 C3IP5D 66779815 IC50 = 1000 nM T94131 CH86MR 66779905 IC50 = 1600 nM T94131 CX2N6E 66779920 IC50 > 790 nM T94131 C9O4TC 66779989 IC50 = 400 nM T94131 CF2UM8 66780001 IC50 = 4000 nM T94131 CHU0C5 66780007 IC50 = 500 nM T94131 CGL4V1 66780016 IC50 = 2000 nM T94131 C5F6OA 66780027 IC50 = 6300 nM T94131 C8DN7A 66780034 IC50 = 4000 nM T94131 C4AM6R 66780100 IC50 = 1300 nM T94131 CZ5P2N 66780118 IC50 = 160 nM T94131 CREA54 66780266 IC50 = 1300 nM T94131 CRCA72 66780292 IC50 = 2500 nM T94131 CW2SM6 66780337 IC50 = 250 nM T94131 CU54DY 66780379 IC50 = 2500 nM T94131 CQ70YA 66780434 IC50 > 7900 nM T94131 C8F9UY 66780515 IC50 = 250 nM T94131 CFH6C2 66780644 IC50 = 2500 nM T94131 CTZB46 66780835 IC50 = 7900 nM T94131 CEP5A2 66780844 IC50 > 6300 nM T94131 C51ARE 66788835 Ki = 5.3 nM T94131 C3PL1S 66800530 IC50 = 63.1 nM T94131 CJN4M2 66806967 IC50 = 630.96 nM T94131 CW12XO 66882257 IC50 > 10000 nM T94131 C6IO1S 66883557 IC50 > 10000 nM T94131 C1HSE0 67035086 IC50 = 980 nM T94131 C38RGB 67035556 IC50 > 9100 nM T94131 C5E4AJ 67050504 IC50 = 11 nM T94131 CMWO25 67061712 IC50 = 1.4 nM T94131 C0OX5N 67103709 IC50 = 1500 nM T94131 C9J2EO 67103712 IC50 = 210 nM T94131 CM4W1Y 67103722 IC50 = 2500 nM T94131 C5TYQ3 67103909 IC50 = 140 nM T94131 CVJ49E 67103974 IC50 = 1200 nM T94131 C3VFY7 67104025 IC50 = 3500 nM T94131 CC07KA 67104052 IC50 = 2900 nM T94131 C4Z0HT 67159178 IC50 <= 10000 nM T94131 C7EZW6 67192973 IC50 = 1600 nM T94131 CQHF85 67284779 IC50 = 2010 nM T94131 CT6BX3 67285457 Ki = 16000 nM T94131 C9LI0M 67294297 Ki = 49.1 nM T94131 C5BZ2V 67981475 IC50 = 1000 nM T94131 CK86XZ 67982080 IC50 = 316.23 nM T94131 CS0TY5 67982485 IC50 = 398.11 nM T94131 C9A2RD 67982543 IC50 = 3981.07 nM T94131 C7A0GH 67982639 IC50 = 1584.89 nM T94131 CW79LA 67982712 IC50 = 1258.93 nM T94131 CEG3F8 67983123 IC50 = 3000 nM T94131 C25AHY 67984037 IC50 = 8500 nM T94131 C7N4ZS 68034365 IC50 = 2400 nM T94131 CG53JO 68044823 Ki = 11 nM T94131 CGA82Q 68044837 Ki = 35 nM T94131 C4RLP9 68044907 Ki = 9 nM T94131 C6U8RP 68045063 Ki = 8 nM T94131 C0LQN1 68045070 Ki = 60 nM T94131 C7DL6V 68045162 Ki = 28 nM T94131 CA4JF3 68045179 Ki = 7 nM T94131 C57DTK 68045182 Ki = 4 nM T94131 CUQ2W1 68095924 IC50 = 158.49 nM T94131 CUR8N0 68096082 IC50 = 501.19 nM T94131 C8I7GC 68293638 IC50 > 10000 nM T94131 C45TIJ 69489467 Ki = 59.8 nM T94131 C8MTV6 70674592 IC50 = 280 nM T94131 CXB45Q 70674939 IC50 = 108 nM T94131 CAR46Z 70675172 IC50 = 72 nM T94131 CN09DI 70675846 IC50 = 97400 nM T94131 C6BQE1 70681248 IC50 = 1600 nM T94131 CPE36T 70681262 IC50 = 200 nM T94131 CPX41V 70682086 IC50 = 6.31 nM T94131 CZ5TI9 70682135 IC50 = 5120 nM T94131 CQW54O 70682591 Ki = 230 nM T94131 CPV59G 70682592 Ki = 1140 nM T94131 CB3ZN5 70683337 IC50 = 2500 nM T94131 C1I5PH 70683338 IC50 = 250 nM T94131 CSM0A6 70684204 IC50 = 2.512 nM T94131 CXD08N 70684690 Ki = 61 nM T94131 CG95EC 70684794 Ki = 84 nM T94131 C8O2QH 70685440 IC50 = 500 nM T94131 CZG9M1 70685441 IC50 = 2000 nM T94131 CH7KO0 70685442 IC50 = 1300 nM T94131 C6G4WB 70686339 IC50 = 251.19 nM T94131 CON8X4 70686340 IC50 = 63.1 nM T94131 C1ASW4 70686341 IC50 = 25.12 nM T94131 C0PWL5 70686455 IC50 = 125.89 nM T94131 CN4CR2 70686584 IC50 = 4100 nM T94131 C85FWA 70686829 Ki = 110 nM T94131 CQS8G7 70686830 Ki = 530 nM T94131 C8QSD2 70688455 IC50 = 7.943 nM T94131 CFCJ02 70688558 IC50 = 15.85 nM T94131 CSX6I7 70688908 Ki = 110 nM T94131 C1U5FC 70689024 Ki = 124 nM T94131 C5YN6U 70689166 IC50 = 5000 nM T94131 C6L4WY 70689639 IC50 = 790 nM T94131 CGT1X2 70690496 IC50 = 25.12 nM T94131 CTY78N 70690549 IC50 = 5740 nM T94131 CW3U5J 70690994 Ki = 260 nM T94131 CC6I1Q 70691259 IC50 = 3200 nM T94131 CD3JL4 70691776 IC50 = 500 nM T94131 CDK52M 70692650 IC50 = 15.85 nM T94131 CGQJ68 70692914 IC50 = 7.943 nM T94131 C7G5UV 70692915 IC50 = 7.943 nM T94131 C3TM1F 70693128 Ki = 57 nM T94131 C2VAU8 70693129 Ki = 32 nM T94131 CU3WF2 70693248 Ki = 26.7 nM T94131 C65FHO 70694723 Ki = 62.9 nM T94131 CPFO83 70694805 IC50 = 12.59 nM T94131 CRNY76 70695188 Ki = 62 nM T94131 C3N5YJ 70695189 Ki = 5810 nM T94131 C75YGN 70695469 IC50 > 3200 nM T94131 C61CFG 70696737 IC50 = 31.62 nM T94131 C7KL5X 70696852 IC50 = 125.89 nM T94131 CRH8E2 71270723 IC50 = 501.19 nM T94131 CWR58A 71270783 IC50 > 1479.11 nM T94131 CF9LU4 71270807 IC50 = 501.19 nM T94131 C7FDL2 71270817 IC50 = 398.11 nM T94131 CNR1G9 71270824 IC50 = 2511.89 nM T94131 C38LBA 71270831 IC50 = 316.23 nM T94131 CTL6R5 71270836 IC50 = 398.11 nM T94131 CM4LX7 71270848 IC50 > 6309.57 nM T94131 C2GWX6 71270906 IC50 = 1995.26 nM T94131 CX0DL3 71270910 IC50 > 3981.07 nM T94131 C0COW6 71270913 IC50 > 6309.57 nM T94131 CB0S8G 71270927 IC50 = 251.19 nM T94131 C24IOW 71270948 IC50 > 5011.87 nM T94131 C5BJ2Y 71270957 IC50 > 3162.28 nM T94131 C03NFY 71271625 IC50 > 5011.87 nM T94131 CL47JU 71271739 IC50 > 7943.28 nM T94131 CS5JG6 71271910 IC50 > 6309.57 nM T94131 C4PSK8 71271965 IC50 = 316.23 nM T94131 CB4N1M 71272066 IC50 > 5011.87 nM T94131 CD8E1Y 71272453 IC50 = 630.96 nM T94131 C8EW9V 71272757 IC50 = 3162.28 nM T94131 C0LO8I 71272765 IC50 = 398.11 nM T94131 C1MVL0 71273460 Ki = 40.6 nM T94131 CK58RV 71449587 IC50 = 91 nM T94131 C0ROQ6 71450451 IC50 = 22 nM T94131 CTL30H 71450452 IC50 = 12 nM T94131 CNX18D 71450453 IC50 = 24 nM T94131 C7HT4F 71450454 IC50 = 46 nM T94131 CNHJ63 71451228 IC50 = 777 nM T94131 CD8Y3S 71451617 Ki = 2350 nM T94131 C9SC2V 71452282 IC50 = 16 nM T94131 CY62VF 71452283 IC50 = 181 nM T94131 CQ7C5R 71452284 IC50 = 14 nM T94131 C6VF7J 71453206 IC50 = 63 nM T94131 CR84JX 71453419 Ki = 4 nM T94131 CZ61FJ 71454160 IC50 = 25.12 nM T94131 CZ8Q5P 71454238 Ki = 2.4 nM T94131 CF74SL 71454944 IC50 = 93 nM T94131 CO82IY 71455167 Ki = 21 nM T94131 CA7L1Y 71455168 Ki = 31 nM T94131 CSW47K 71455817 IC50 = 117 nM T94131 CT32GB 71455818 IC50 = 10 nM T94131 CE1IX7 71456728 IC50 = 59 nM T94131 CLUR84 71457607 IC50 = 12 nM T94131 C4ACV9 71457608 IC50 = 95 nM T94131 CM1ND2 71458573 IC50 = 82 nM T94131 C3S0NP 71458574 IC50 = 72 nM T94131 CY6WI2 71458575 IC50 = 60 nM T94131 C13KJV 71459500 IC50 = 250 nM T94131 CO8U5R 71459501 IC50 = 223 nM T94131 CL30DJ 71459502 IC50 = 346 nM T94131 C1Y8WD 71459503 IC50 = 12 nM T94131 CT7K3A 71460422 IC50 = 54 nM T94131 CW9YM2 71461240 IC50 = 3 nM T94131 CA2V9S 71461241 IC50 = 161 nM T94131 C65RJY 71461242 IC50 = 25 nM T94131 C2HOB7 71461243 IC50 = 3 nM T94131 CO26VM 71462973 IC50 = 24 nM T94131 CU3EO6 71520393 IC50 > 10000 nM T94131 CYC6S1 71520394 IC50 > 10000 nM T94131 C1KMX0 71520395 IC50 > 10000 nM T94131 CYK7N8 71520396 IC50 > 10000 nM T94131 CTC0O8 71520397 IC50 > 10000 nM T94131 C0UZ3D 71526877 IC50 = 2000 nM T94131 CP05SQ 71526878 IC50 = 100000 nM T94131 CZK6X9 71526879 IC50 > 10000 nM T94131 C8QRE4 71526880 IC50 > 10000 nM T94131 CT3QI8 71526881 IC50 > 10000 nM T94131 CO4MY1 71527005 IC50 > 10000 nM T94131 CJC64F 71527006 IC50 > 10000 nM T94131 C96WZG 71527007 IC50 = 3900 nM T94131 CUC7I1 71527008 IC50 = 8000 nM T94131 C09WKC 71527009 IC50 > 10000 nM T94131 CSPO76 71527716 IC50 > 5011.87 nM T94131 CIN7O1 71527842 IC50 > 6309.57 nM T94131 CO6CI7 71528725 IC50 = 9900 nM T94131 C5U2ZC 71528726 IC50 = 380 nM T94131 CTKO36 71528727 IC50 = 3600 nM T94131 C2KF3X 71533728 IC50 = 1046 nM T94131 CI7Q4K 71548718 IC50 = 2700 nM T94131 CED62L 71548719 IC50 = 9200 nM T94131 C4B0KN 71549093 IC50 = 20000 nM T94131 C6PRV1 71655831 IC50 = 12 nM T94131 CU48RN 71657825 IC50 = 154 nM T94131 CWG8M3 71682651 IC50 = 210 nM T94131 C6UGW3 71682652 IC50 = 4600 nM T94131 C7BX4K 71682653 IC50 = 930 nM T94131 CQX8N3 71682654 IC50 > 10000 nM T94131 CS32HB 71716798 IC50 > 6309.57 nM T94131 C07GCV 71716799 IC50 = 5011.87 nM T94131 CFW01E 71718034 IC50 = 2530 nM T94131 CXJC41 72188489 IC50 = 1000 nM T94131 C29KOU 72709209 IC50 > 10000 nM T94131 CT73IW 72709284 IC50 = 2500 nM T94131 CIL6S8 72737375 IC50 = 28 nM T94131 CTYJ25 72737376 IC50 = 158 nM T94131 CPL27S 72737377 IC50 = 52 nM T94131 C5RQB7 72737378 IC50 = 68 nM T94131 C8H7VT 72737379 IC50 = 121 nM T94131 CV2G1F 72737380 IC50 = 62 nM T94131 CHX84Q 72737381 IC50 = 7.2 nM T94131 CI5OT1 72737382 IC50 = 203 nM T94131 CSN5U8 72737551 IC50 = 17 nM T94131 CHC5J2 72737552 IC50 = 29 nM T94131 CB5PM9 72737553 IC50 = 68 nM T94131 CIF36E 72737554 IC50 = 57 nM T94131 C87HDL 72737555 IC50 = 100 nM T94131 CVU2J9 72949025 IC50 = 42 nM T94131 CC6KY3 72949203 IC50 = 16 nM T94131 CYGV85 73051332 IC50 = 5 nM T94131 CV4BH5 73051810 IC50 = 34 nM T94131 CE2IG4 73051811 IC50 = 271 nM T94131 CKUF15 73051812 IC50 = 4 nM T94131 CRF25X 73051813 IC50 = 12 nM T94131 C56JVH 73051977 IC50 = 67 nM T94131 C7N0AF 73052137 IC50 = 11 nM T94131 CNTD65 73052455 IC50 = 6 nM T94131 CZY9U8 73441896 IC50 = 31622.78 nM T94131 CL0XZ1 73659199 Ki = 2 nM T94131 CK7XM5 73659200 Ki = 1 nM T94131 C8EI1X 73673707 IC50 = 1.5 nM T94131 C0W1TK 73774799 IC50 = 120 nM T94131 C4W3IL 73774944 IC50 = 420 nM T94131 CH75QS 73774946 IC50 = 11 nM T94131 C5NKS4 73774948 IC50 = 40 nM T94131 C23MSN 73775105 IC50 = 160 nM T94131 CQG43I 73775546 IC50 = 3.3 nM T94131 CBXV38 73775549 IC50 = 3.1 nM T94131 C6O4PV 73775675 IC50 = 15 nM T94131 CQI4G9 73775798 IC50 = 81 nM T94131 CG0VK1 73775800 IC50 = 17 nM T94131 C7N0ME 73775931 IC50 = 3.6 nM T94131 CA5DJ3 73775934 IC50 = 13 nM T94131 CD6M4Q 73776065 IC50 = 10 nM T94131 C6X3LA 73776070 IC50 = 0.3 nM T94131 C5PKH6 73776209 IC50 = 430 nM T94131 C4WLT1 73776507 IC50 = 12 nM T94131 CPH39S 73776508 IC50 = 45 nM T94131 CT6ZB1 73776511 IC50 = 64 nM T94131 CI9K0J 73776652 IC50 = 0.7 nM T94131 CMHK83 73776786 IC50 = 0.6 nM T94131 CMT13V 73776787 IC50 = 6.8 nM T94131 CBYN18 73977439 IC50 = 1995 nM T94131 C9V1YR 73977449 IC50 = 251 nM T94131 CXA90D 73977451 IC50 = 316 nM T94131 CEZ7L2 73977461 IC50 = 126 nM T94131 CD0T9V 74539799 IC50 = 0.74 nM T94131 C16KOS 74539862 IC50 = 1.1 nM T94131 CN2MI8 76310247 IC50 > 50000 nM T94131 CKO41J 76310248 IC50 = 741 nM T94131 CEN9Q5 76310249 IC50 > 50000 nM T94131 CJCF67 76310250 IC50 = 26 nM T94131 CBF70W 76310805 IC50 = 316.23 nM T94131 CA2VR6 76311340 IC50 = 194.98 nM T94131 CMR07I 76313939 IC50 > 50000 nM T94131 C5P2CJ 76313940 IC50 = 30700 nM T94131 CAV5Q9 76313941 IC50 = 22000 nM T94131 CO13XZ 76314937 IC50 = 386 nM T94131 C7W2HI 76314938 IC50 = 341.98 nM T94131 C6H9EL 76314939 IC50 = 230.99 nM T94131 C0J6PL 76317466 IC50 > 50000 nM T94131 CVW35P 76317467 IC50 > 50000 nM T94131 CZ1T3C 76317468 IC50 > 50000 nM T94131 C4MKN3 76317469 IC50 = 62 nM T94131 C3JA4F 76317470 IC50 = 353 nM T94131 C4XJ5Y 76317471 IC50 = 153 nM T94131 CS6ME5 76318566 IC50 = 235 nM T94131 CG4I2R 76318567 IC50 = 217 nM T94131 C8E4GI 76321204 IC50 = 183 nM T94131 CF4OI8 76321205 IC50 = 12300 nM T94131 C1YFK9 76322218 IC50 = 267.98 nM T94131 CL0T7B 76322219 IC50 <= 65 nM T94131 CDG8V4 76324821 IC50 = 87 nM T94131 CJW39V 76324822 IC50 > 50000 nM T94131 C2BFA1 76324823 IC50 = 4700 nM T94131 CM4N8A 76325342 IC50 = 6309.57 nM T94131 C92ZAB 76325343 IC50 = 25118.86 nM T94131 C1HFI9 76325446 IC50 = 3259 nM T94131 C4GZ1Q 76325833 IC50 = 357.03 nM T94131 CQ31CA 76325834 IC50 = 312.97 nM T94131 C4A8XZ 76328376 IC50 = 3400 nM T94131 C39CLE 76329428 IC50 = 247 nM T94131 CYR0G6 76332050 IC50 = 6300 nM T94131 C4MID5 76332051 IC50 = 7880 nM T94131 C70WJE 76332052 IC50 = 79 nM T94131 CQ8YC1 76332568 IC50 = 7.943 nM T94131 CE6BI0 76332666 IC50 = 4350 nM T94131 C16SRX 76333068 IC50 = 143 nM T94131 CW81MC 76333069 IC50 = 264.97 nM T94131 C26CKL 76333070 IC50 = 153.99 nM T94131 C47NLT 76333071 IC50 = 250 nM T94131 CN38BK 76335378 IC50 = 81 nM T94131 C69ATM 76335666 IC50 > 50000 nM T94131 C0SI4C 76335667 IC50 > 50000 nM T94131 C31NEK 76335668 IC50 = 574 nM T94131 CL6BV5 76335669 IC50 > 50000 nM T94131 C73KJD 76335670 IC50 = 227 nM T94131 CY3LO5 76336173 IC50 = 1258.93 nM T94131 CJ3V6Y 76336695 IC50 = 274 nM T94131 CD03GB 76336696 IC50 = 277.97 nM T94131 C2JTH8 77107528 IC50 = 112 nM T94131 C42HDP 77107927 IC50 = 42 nM T94131 C04SRC 77147259 IC50 = 1774 nM T94131 C9I7TY 78319187 IC50 = 1584.89 nM T94131 C24LQH 78320362 IC50 = 35 nM T94131 C9T8KF 78320671 IC50 = 70 nM T94131 CI2YN8 78320672 IC50 = 24 nM T94131 CI6K4J 78320673 IC50 = 305 nM T94131 COFJ16 78320996 IC50 = 5200 nM T94131 CMU5P2 78321310 IC50 = 150 nM T94131 CE13AJ 78321314 IC50 = 200 nM T94131 CSP2H4 78321635 IC50 = 280 nM T94131 CWA0B1 78322567 IC50 = 140 nM T94131 CH6P9D 78322877 IC50 > 10000 nM T94131 C4IW9V 78323193 IC50 = 230 nM T94131 CD1JC8 78324443 IC50 = 129 nM T94131 C04IKP 86268622 IC50 = 28 nM T94131 C5P3RO 86647783 IC50 = 1200 nM T94131 CDXM47 86677874 IC50 > 10000 nM T94131 CP3W1B 86695297 IC50 > 20000 nM T94131 CA17UE 86732669 IC50 = 4630 nM T94131 C2PCS7 87061302 IC50 = 181 nM T94131 CNVS32 87343636 Ki = 16.7 nM T94131 CV6PI8 87562294 IC50 = 125.89 nM T94131 CZ2AU4 87570781 IC50 = 375 nM T94131 C3HD5O 88570842 Ki = 9 nM T94131 CLEX32 89034287 Ki = 4 nM T94131 C1AKZ4 89034365 Ki = 6 nM T94131 CEQ80V 89034380 Ki = 5 nM T94131 C1HB3F 89051931 IC50 = 330 nM T94131 C61SCX 89493851 IC50 = 5 nM T94131 C1LU3X 89493904 IC50 = 31 nM T94131 CTE1L0 89517065 IC50 = 9300 nM T94131 C56KSC 89517226 IC50 > 10000 nM T94131 C6M0QF 89841854 IC50 = 400 nM T94131 C61GIO 89841941 IC50 = 40 nM T94131 C6FI0A 89842032 IC50 = 110 nM T94131 COL45N 89842055 IC50 = 60 nM T94131 C7FNP8 89842123 IC50 = 25 nM T94131 CF50MO 89842136 IC50 = 1100 nM T94131 C6CKP2 89842150 IC50 = 50 nM T94131 CVZH15 89842186 IC50 = 240 nM T94131 C2LQ9V 89842220 IC50 = 150 nM T94131 C83SXM 89842240 IC50 = 1100 nM T94131 CQ1U2Y 89842245 IC50 = 1000 nM T94131 CQO85K 89842249 IC50 > 7000 nM T94131 CX70NQ 89842250 IC50 = 14 nM T94131 CN5Y9A 90064110 IC50 = 27 nM T94131 C7FP2M 90064111 IC50 = 4 nM T94131 CN51BK 90064299 IC50 = 2 nM T94131 CUZ13D 90102336 IC50 = 0.7 nM T94131 CQO9J0 90103194 IC50 = 1.7 nM T94131 C28WQY 90431726 IC50 = 20 nM T94131 C08UWK 90665816 IC50 = 100000 nM T94131 CMWB58 91757958 IC50 <= 10000 nM T94131 C3Y0DS 91801158 IC50 = 2.6 nM T94131 CAS7W6 91864650 IC50 = 8440 nM T94131 CA3ZC1 92172785 IC50 = 575000 nM T94131 C4JMV1 118003503 IC50 = 330 nM T94131 C6YRW7 118003617 IC50 = 110 nM T94131 C8QHY9 118003714 IC50 = 75 nM T94131 CLDA15 118003719 IC50 = 360 nM T94131 C5LW9G 118004010 IC50 = 100 nM T94131 CK0W1T 118004012 IC50 = 170 nM T94131 C0BIP8 118004016 IC50 = 350 nM T94131 CB4PM3 118004022 IC50 = 110 nM T94131 CNCK58 118004064 IC50 = 280 nM T94131 C14WCU 118131317 IC50 > 1000 nM T94131 C67VQE 118341819 IC50 = 850 nM T94131 CC9P5H 118341835 IC50 = 750 nM T94131 CUMA23 118341844 IC50 = 1840 nM T94131 C3IP9X 118341852 IC50 = 190 nM T94131 C6TI0Z 118341865 IC50 = 520 nM T94131 C4U7NC 118341870 IC50 = 360 nM T94131 CVL03K 118341884 IC50 = 1370 nM T94131 CPZN96 118341923 IC50 = 150 nM T94131 C9E3DU 118341927 IC50 = 6950 nM T94131 CVN87P 118433737 IC50 = 36 nM T94131 C8W1RN 118445922 IC50 = 7 nM T94131 CGYA58 118445928 IC50 = 182 nM T94131 CL29BI 118445929 IC50 = 52 nM T94131 CI24WZ 118445978 IC50 = 3 nM T94131 CA20CO 118445983 IC50 = 13 nM T94131 CQF1V4 118446049 IC50 = 4 nM T94131 C90OAT 118446064 IC50 = 43 nM T94131 CJQ92T 118572891 IC50 < 10 nM T94131 CVY45K 118575373 IC50 > 10000 nM T94131 CS20UM 118575423 IC50 > 10000 nM T94131 CCPV26 118575517 IC50 = 632 nM T94131 C0L9JQ 118575526 IC50 = 1300 nM T94131 CH6AB7 118575540 IC50 > 10000 nM T94131 C97QIN 118575555 IC50 = 990 nM T94131 CEDC48 118575654 IC50 = 3466 nM T94131 COYJ84 118575663 IC50 > 10000 nM T94131 CS1Z8W 118575682 IC50 = 4407 nM T94131 CC0S4G 118575689 IC50 = 199 nM T94131 C6X8HG 118575694 IC50 > 10000 nM T94131 CUJ30I 118575784 IC50 = 1247 nM T94131 CAT54V 118575791 IC50 = 1277 nM T94131 C1K6HU 118575835 IC50 = 4262 nM T94131 C2OQ4U 118575893 IC50 > 10000 nM T94131 C6HEA7 118575940 IC50 = 990 nM T94131 CIU7J3 118575971 IC50 = 267 nM T94131 CAD39P 118575986 IC50 = 4150 nM T94131 CCYI54 118576050 IC50 = 1131 nM T94131 CW9T6F 118576060 IC50 = 7836 nM T94131 C7Y4AT 118576103 IC50 > 10000 nM T94131 C47WMX 118576166 IC50 = 7989 nM T94131 C1UT8B 118576192 IC50 > 10000 nM T94131 C0F7JV 118576207 IC50 = 2311 nM T94131 CU61WD 118576212 IC50 > 10000 nM T94131 CE3V8W 118576268 IC50 = 54 nM T94131 CO0YC8 118616775 IC50 = 1 nM T94131 CS5C8W 118684133 IC50 = 4.3 nM T94131 CRX24W 118709077 IC50 = 6000 nM T94131 CV2EJ7 118709081 IC50 = 6900 nM T94131 CZ41AQ 118709092 IC50 = 83000 nM T94131 CR6ML1 118709578 IC50 = 670 nM T94131 C0OH7I 118709579 IC50 = 13500 nM T94131 C73YIO 118709582 IC50 = 3000 nM T94131 CGWX02 118709583 IC50 = 510 nM T94131 CY2QG0 118711873 IC50 = 10890 nM T94131 CH4XY2 118711874 IC50 = 10710 nM T94131 C94GZM 118712046 IC50 = 3600 nM T94131 CPXQ86 118721834 Ki = 44 nM T94131 CH9D8G 118721835 Ki = 19 nM T94131 CYHG95 118721836 Ki = 21 nM T94131 CP6SR7 118721837 Ki = 9 nM T94131 CW4N7Q 118721838 Ki = 7 nM T94131 CZG78A 118721839 Ki = 190 nM T94131 C2BQS3 118721840 Ki = 6 nM T94131 C2T9RN 118721841 Ki = 1 nM T94131 C6GJ0Q 118721842 Ki = 7 nM T94131 C9RPN4 118721843 Ki = 2 nM T94131 CYNZ53 118721844 Ki = 22 nM T94131 C5R1VP 118721845 Ki = 19 nM T94131 CB53EU 118728320 IC50 = 34624 nM T94131 C6KJL1 118728321 IC50 = 21668 nM T94131 CKJ3S6 118728322 IC50 = 27916 nM T94131 CT0L3Y 118728325 IC50 = 24342 nM T94131 CHS2E4 118728326 IC50 = 11812 nM T94131 CRUP47 118728328 IC50 = 44117 nM T94131 CQR41G 118728330 IC50 = 19479 nM T94131 CN4Q9R 118728332 IC50 = 9443 nM T94131 CDI10F 118728336 IC50 = 41626 nM T94131 CHT6K9 118728811 Ki = 2900 nM T94131 CUA3Y2 118728812 Ki > 4000 nM T94131 CDQ78G 118728813 Ki = 400 nM T94131 CZ6XL7 118728814 Ki = 630 nM T94131 CMO67K 118728815 Ki = 750 nM T94131 CR2M0Q 118728816 Ki = 1500 nM T94131 C62SCL 118728817 Ki = 690 nM T94131 CSB30C 118728819 Ki = 1100 nM T94131 CV7XU8 118728820 Ki = 710 nM T94131 C3J1EX 118728821 Ki > 4000 nM T94131 CIWB78 118728822 Ki > 4000 nM T94131 CP18SE 118728823 Ki = 780 nM T94131 CM42CA 118728824 Ki = 1400 nM T94131 C9Q7CL 118728825 Ki = 2800 nM T94131 CCR3S0 118728826 Ki = 1200 nM T94131 CB1WC5 118729946 IC50 = 380 nM T94131 CQ4G9M 118729947 IC50 = 1600 nM T94131 C43IPJ 118729948 IC50 = 250 nM T94131 C3I9CQ 118729949 IC50 = 510 nM T94131 CZQ17M 118729950 IC50 = 200 nM T94131 C3G1ZP 118729951 IC50 = 4950 nM T94131 CY60FC 118730033 IC50 = 17087 nM T94131 CN3B4U 118730711 IC50 = 320 nM T94131 C0IL3N 118730712 IC50 = 1400 nM T94131 C3CH1A 118730713 IC50 = 350 nM T94131 CHX5L9 118730714 IC50 = 250 nM T94131 CNJ32C 118730715 IC50 = 3200 nM T94131 C1MKB3 118730716 IC50 = 1400 nM T94131 C81RJA 118730717 IC50 = 13000 nM T94131 CFZ16R 118737301 IC50 <= 10000 nM T94131 C27CPQ 118737302 IC50 <= 10000 nM T94131 C59VXA 118737303 IC50 <= 10000 nM T94131 CGO1N4 118737304 IC50 <= 10000 nM T94131 CS85FM 118737305 IC50 <= 10000 nM T94131 C8UCO1 118737306 IC50 <= 10000 nM T94131 CR0BZ2 118737307 IC50 <= 10000 nM T94131 C3N4DJ 118737308 IC50 <= 10000 nM T94131 CGY5B1 118737309 IC50 <= 10000 nM T94131 CV85EL 118981804 IC50 = 38 nM T94131 C91PVZ 121428416 IC50 = 204 nM T94131 CA2DM0 121428489 IC50 = 164 nM T94131 CQLX36 121428567 IC50 = 288 nM T94131 CFN12W 121445751 IC50 = 28 nM T94131 C04NDW 121445810 IC50 = 41 nM T94131 C81IFQ 122163152 IC50 = 1340 nM T94131 C2VGD5 122178120 IC50 = 21.1 nM T94131 C24XUZ 122178124 IC50 = 10.2 nM T94131 CN5AB3 122179486 IC50 = 4.4 nM T94131 CLEK13 122179487 IC50 = 10 nM T94131 C0OW8H 122179490 IC50 = 52 nM T94131 C0VD5F 122179491 IC50 = 2 nM T94131 CQ87FB 122179492 IC50 = 4 nM T94131 CBJ29X 122179493 IC50 > 10000 nM T94131 CA5N1B 122179494 IC50 = 25 nM T94131 CM4AW9 122180514 Ki = 0.024 nM T94131 CM89OL 122180515 Ki = 0.016 nM T94131 CU0C1D 122180516 Ki = 0.01 nM T94131 CB6PR7 122180517 Ki = 0.034 nM T94131 CQ63DW 122180518 Ki = 0.006 nM T94131 C9N8JT 122180519 Ki = 0.003 nM T94131 C42GSX 122180520 Ki = 0.002 nM T94131 CVA3P2 122180521 Ki = 0.009 nM T94131 C0A7CQ 122180522 Ki = 0.025 nM T94131 CEFS13 122180793 IC50 = 91560 nM T94131 CFZ2E1 122180794 IC50 = 125800 nM T94131 C5YKG7 122180795 IC50 = 465500 nM T94131 C9ID7U 122180796 IC50 = 345900 nM T94131 C08XOC 122180839 IC50 = 781500 nM T94131 C2HM6P 122180840 IC50 = 967700 nM T94131 CT9Y6U 122180841 IC50 = 23640 nM T94131 C6FOM0 122180842 IC50 = 18480 nM T94131 COX90L 122180843 IC50 = 12570 nM T94131 CP40RU 122180844 IC50 = 26870 nM T94131 CC0EK9 122180845 IC50 = 15560 nM T94131 CS85CU 122181413 IC50 = 280 nM T94131 CQS67B 122181416 IC50 = 650 nM T94131 C58XRY 122184465 IC50 = 1995.26 nM T94131 C16ALM 122184466 IC50 = 1000 nM T94131 CDZY02 122184468 IC50 = 50118.72 nM T94131 CTH70U 122184469 IC50 = 12589.25 nM T94131 C9ZXR7 122184470 IC50 = 3981.07 nM T94131 CNJ9Z4 122184471 IC50 = 3981.07 nM T94131 CS41EG 122184473 IC50 = 1258.93 nM T94131 CZ36GL 122184474 IC50 = 1000 nM T94131 CU4ZT6 122184475 IC50 = 10000 nM T94131 C3H9PR 122184476 IC50 = 1258.93 nM T94131 CU40TW 122184477 IC50 = 3162.28 nM T94131 CAMD31 122184479 IC50 = 19952.62 nM T94131 C1F9RK 122184480 IC50 = 251.19 nM T94131 C7XW1K 122184481 IC50 = 12589.25 nM T94131 CRUX54 122184482 IC50 = 31622.78 nM T94131 CQ7W0P 122184526 IC50 = 3981.07 nM T94131 CA5YB2 122184529 IC50 = 2511.89 nM T94131 C64YPH 122184530 IC50 = 2511.89 nM T94131 C4AGX5 122184531 IC50 = 3162.28 nM T94131 CQL4K5 122184532 IC50 = 1584.89 nM T94131 CRKV74 122184533 IC50 = 3981.07 nM T94131 CX14YD 122184534 IC50 = 1000 nM T94131 CM6A4S 122184535 IC50 = 1258.93 nM T94131 CF86YS 122184536 IC50 = 1995.26 nM T94131 CYRH97 122184538 IC50 = 3162.28 nM T94131 CD4W0Z 122184539 IC50 = 10000 nM T94131 CH8Y3Q 122184540 IC50 = 15848.93 nM T94131 CDA85R 122184541 IC50 = 63095.73 nM T94131 CF36XJ 122184542 IC50 > 199526.23 nM T94131 CQ6O7H 122184543 IC50 = 50118.72 nM T94131 CS4MN0 122184544 IC50 = 10000 nM T94131 CKT74G 122185265 IC50 = 14 nM T94131 CJ6C1O 122185267 IC50 = 22 nM T94131 CGW35U 122387497 IC50 = 259 nM T94131 C38BML 122387499 IC50 = 265 nM T94131 CCW0M1 122387500 IC50 = 174 nM T94131 CKA90Y 122387501 IC50 = 89 nM T94131 CH4LC6 122387502 IC50 = 56 nM T94131 C8OC3E 122387504 IC50 = 169 nM T94131 C34AHY 122387505 IC50 = 185 nM T94131 CUG1T6 122387506 IC50 = 98 nM T94131 CE7K5C 122387507 IC50 = 173 nM T94131 C4HL3N 122387508 IC50 = 111 nM T94131 CA7L3S 122387509 IC50 = 112 nM T94131 CR9NF3 122542400 IC50 = 5.7 nM T94131 CZE35C 122648343 IC50 > 10000 nM T94131 C54RNT 122648367 IC50 > 10000 nM T94131 C1UVI7 122648600 IC50 = 255 nM T94131 CMX59K 122648648 IC50 = 8.1 nM T94131 CVZ64I 122648649 IC50 > 10000 nM T94131 CPTY78 124518210 IC50 = 89 nM T94131 CB7G5E 126476620 IC50 = 501.19 nM T94131 C74BNR 126480568 IC50 = 1584.89 nM T94131 C1N6YP 126480569 IC50 = 2511.89 nM T94131 CE52HC 126480570 IC50 = 630.96 nM T94131 CQ74WU 126480571 IC50 = 3981.07 nM T94131 C0AFE2 126480572 IC50 = 1000 nM T94131 C3E7JB 126480573 IC50 = 6309.57 nM T94131 CPW54V 126480574 IC50 = 1000 nM T94131 CVJ3Q5 127025094 IC50 = 285 nM T94131 C2E4LO 127025141 IC50 = 6570 nM T94131 CO94KJ 127025144 IC50 > 25000 nM T94131 CKO53P 127025146 IC50 = 21450 nM T94131 CF7H0V 127025161 IC50 = 1260 nM T94131 CE4C3J 127025163 IC50 = 12360 nM T94131 CAV24Z 127025164 IC50 = 9360 nM T94131 C98DKI 127025346 IC50 = 4 nM T94131 CDZ56M 127025449 IC50 > 25000 nM T94131 CBXJ67 127025628 IC50 = 2.7 nM T94131 CH2Q7A 127027634 IC50 = 280 nM T94131 CSV3R7 127029064 IC50 = 64 nM T94131 CQTG79 127029604 IC50 = 279 nM T94131 CZHT45 127031017 IC50 = 3700 nM T94131 CU0F4R 127031332 IC50 = 1500 nM T94131 C2IN4Q 127031333 IC50 > 50000 nM T94131 CS12RU 127031435 IC50 = 2.3 nM T94131 CGU4H3 127031891 IC50 = 21 nM T94131 CGKR53 127032915 IC50 = 502 nM T94131 C41YQI 127035981 IC50 = 939 nM T94131 C7V4WA 127036623 IC50 = 13780 nM T94131 CJ1LH4 127036935 IC50 = 3120 nM T94131 CG8DA9 127045861 IC50 = 99 nM T94131 CVF8Z9 127045862 IC50 = 5 nM T94131 CH68NT 127046076 IC50 = 77 nM T94131 CA2XD5 127046077 IC50 = 230 nM T94131 COJ68G 127046117 IC50 = 1900 nM T94131 C34REM 127046317 IC50 = 570 nM T94131 CC4ND8 127046862 IC50 = 302 nM T94131 CY2P1X 127047138 IC50 = 440 nM T94131 CZ2R0C 127047140 IC50 = 120 nM T94131 CT89GI 127047683 IC50 = 720 nM T94131 C7D0FN 127047685 IC50 = 240 nM T94131 CN94CQ 127047797 IC50 = 140 nM T94131 C3IC2Z 127052212 IC50 = 5803 nM T94131 CN9XL1 129262531 IC50 = 90 nM T94131 CW7A5X 129626595 IC50 = 3981.07 nM T94131 C18NHD 130302549 IC50 <= 10000 nM T94131 CL13RZ 130302558 IC50 <= 10000 nM T94131 CF5JZ3 130302563 IC50 <= 10000 nM T94131 CD46EL 130302605 IC50 <= 10000 nM T94131 CNI8M6 130302620 IC50 <= 10000 nM T94131 CI6WN9 130302651 IC50 <= 10000 nM T94131 C5ZP0L 130302658 IC50 <= 10000 nM T94131 CW61SG 130302663 IC50 <= 10000 nM T94131 CB27ZG 130302668 IC50 <= 10000 nM T94131 C5VYM6 130302674 IC50 <= 10000 nM T94131 C0FQR2 130302675 IC50 <= 10000 nM T94131 CB34HQ 130302676 IC50 <= 10000 nM T94131 CQR1I8 130302685 IC50 <= 10000 nM T94131 C17DZF 130302698 IC50 <= 10000 nM T94131 CBC6W7 130302701 IC50 <= 10000 nM T94131 CBT21G 130302702 IC50 <= 10000 nM T94131 CDZ45O 130302703 IC50 <= 10000 nM T94131 C2GWU8 130302709 IC50 <= 10000 nM T94131 CV3M6Y 130302710 IC50 <= 10000 nM T94131 C39UQN 130302731 IC50 <= 10000 nM T94131 CL9O8X 130302732 IC50 <= 10000 nM T94131 CL69GM 130302740 IC50 <= 10000 nM T94131 CH8YK9 130302741 IC50 <= 10000 nM T94131 CQR2W9 130302781 IC50 <= 10000 nM T94131 C9HC8A 130302803 IC50 <= 10000 nM T94131 CIK25W 130302809 IC50 <= 10000 nM T94131 CI08PF 130332501 IC50 <= 10000 nM T94131 C1H4UT 130332505 IC50 <= 10000 nM T94131 CZPI64 130332579 IC50 <= 10000 nM T94131 CDS9F3 130332582 IC50 <= 10000 nM T94131 C3G0HF 130332585 IC50 <= 10000 nM T94131 CX13UC 130332620 IC50 <= 10000 nM T94131 CED6F3 130332657 IC50 <= 10000 nM T94131 C73KWM 130338615 IC50 = 100 nM T94131 CLC06T 130406587 IC50 = 1 nM T94131 C47CAY 130421765 IC50 = 0.631 nM T94131 C84YKI 130422161 IC50 = 0.7943 nM T94131 C2MVE6 130422162 IC50 = 0.631 nM T94131 CK68CA 130453737 IC50 = 3000 nM T94131 CUO41K 130470684 IC50 = 7100 nM T94131 CDE7T3 132005217 IC50 = 49 nM T94131 CL26YS 132005219 IC50 = 310 nM T94131 CP32GB 132005220 IC50 = 15 nM T94131 CG1NC4 132005221 IC50 = 3300 nM T94131 C0UV2M 132005224 IC50 = 58 nM T94131 CUN18W 132005225 IC50 = 6.5 nM T94131 CD84OI 132005228 IC50 = 2.8 nM T94131 C9VDI0 132005229 IC50 = 110 nM T94131 CB1Z7P 132005231 IC50 = 340 nM T94131 C7ASP9 132005246 IC50 = 11 nM T94131 C8VE6T 132005248 IC50 = 560 nM T94131 C7LCW1 132005249 IC50 = 110 nM T94131 C5W9LN 132005323 IC50 = 120 nM T94131 CQ6GO2 132005326 IC50 = 330 nM T94131 C6OXE3 132134663 IC50 = 10 nM T94131 C4M8WN 132209922 IC50 = 1.3 nM T94131 CFI23B 132210082 IC50 = 21 nM T94131 C8RK4V 132218631 IC50 = 300 nM T94131 CZD9F3 132219135 IC50 > 10000 nM T94131 CH8DP7 132220479 IC50 = 41 nM T94131 C4Q5LF 132471857 IC50 = 10 nM T94131 CJE34F 132597748 IC50 = 3220 nM T94131 CCV46G 132606879 IC50 = 199.53 nM T94131 CT2PN8 132990561 IC50 = 75 nM T94131 CFG90E 134132909 IC50 = 642 nM T94131 CI49TK 134133218 IC50 = 65 nM T94131 C4YNH0 134134126 IC50 = 698 nM T94131 C0EK8P 134134680 IC50 = 828 nM T94131 C0A1UM 134138053 IC50 = 282 nM T94131 CQ2S4X 134138703 IC50 > 9100 nM T94131 CL3Q6G 134140420 IC50 = 1210 nM T94131 CDJ10M 134142931 IC50 = 1230 nM T94131 CUE85S 134143151 IC50 > 50000 nM T94131 CQ9G7H 134145670 IC50 = 220 nM T94131 C6G8EJ 134146051 IC50 = 40000 nM T94131 CIPL93 134147099 IC50 = 2070 nM T94131 C8ITR3 134147904 IC50 > 50000 nM T94131 CXA3V0 134148445 IC50 = 3780 nM T94131 CXU92M 134150578 IC50 = 366 nM T94131 CG8LE2 134151667 IC50 < 10000 nM T94131 CK43EY 134152988 IC50 = 2940 nM T94131 CS2QP7 134154582 IC50 = 194 nM T94131 C2QGB3 134156160 IC50 = 978 nM T94131 C42RJH 134157534 IC50 = 5859 nM T94131 C9C3XT 134163708 IC50 = 0.631 nM T94131 CD9ZR6 134372929 IC50 = 440 nM T94131 CCS6I3 134372959 IC50 = 4156 nM T94131 CTD03Q 134611885 IC50 >= 199.53 nM T94131 CJXA12 134611894 IC50 <= 0.7943 nM T94131 CX0UR7 134694318 IC50 > 1000 nM T94131 C6LYD2 135121892 IC50 = 63.1 nM T94131 C9FUK2 135151360 IC50 = 52 nM T94131 CT0GQ6 135197577 IC50 = 1.7 nM T94131 C87VKA 135197594 IC50 = 0.93 nM T94131 C0YK5W 135197617 IC50 = 1.6 nM T94131 CF6DJ2 135197621 IC50 = 2.1 nM T94131 CDT25A 135197623 IC50 = 1.5 nM T94131 CQXS07 135197635 IC50 = 1.2 nM T94131 C7KXF1 135197643 IC50 = 1.3 nM T94131 CY38TL 135391000 IC50 = 89.7 nM T94131 COG86Z 135397763 IC50 = 3162.28 nM T94131 CWL67T 135397764 IC50 = 1000 nM T94131 CX8AI4 135398491 IC50 = 180 nM T94131 CQN49C 135409495 IC50 = 4000 nM T94131 C6AZ2R 135435018 IC50 > 25118.86 nM T94131 CMGY62 135485500 IC50 = 273 nM T94131 CM9NV6 135492341 IC50 = 1200 nM T94131 CWJQ64 135492555 IC50 = 968 nM T94131 C3QJ8W 135566371 IC50 = 20 nM T94131 C24ZGX 135566644 IC50 > 10000 nM T94131 C2QDV5 135566741 IC50 > 10000 nM T94131 CTJ6B2 135610083 IC50 = 5900 nM T94131 CN2ME4 135610084 IC50 = 4700 nM T94131 C4G6JF 135610087 IC50 = 5100 nM T94131 CPV59N 135685787 Ki = 1000 nM T94131 C2UN0D 135742360 IC50 > 83300 nM T94131 CI98OY 135750190 IC50 = 195 nM T94131 CF0VL3 135750206 IC50 = 48000 nM T94131 CY4CZ0 135750219 IC50 = 1300 nM T94131 CU29YK 135750268 IC50 = 680 nM T94131 C02PHA 135927892 IC50 > 25118.86 nM T94131 CS8T3D 135927897 IC50 = 5011.87 nM T94131 CF1PS8 135934877 Ki = 1300 nM T94131 C12UDA 135947972 IC50 = 187 nM T94131 CN42ZS 135947973 IC50 = 1500 nM T94131 CF8AO3 135947974 IC50 = 118 nM T94131 CW08GJ 135947976 IC50 = 89 nM T94131 C8O9HG 135947977 IC50 = 50000 nM T94131 CJN7E2 135947978 IC50 = 190 nM T94131 CFKH34 135947979 IC50 = 587 nM T94131 C58FHM 135961523 IC50 = 6918.31 nM T94131 CTRL59 135976660 Ki = 540 nM T94131 C9OAV5 135986100 IC50 = 100000 nM T94131 C3USL8 135986101 IC50 > 100000 nM T94131 C4G2HP 135995897 IC50 = 5780 nM T94131 CNF15Q 135995898 IC50 = 1340 nM T94131 C98HZG 135995899 IC50 = 7640 nM T94131 CIQ82W 135995900 IC50 = 4560 nM T94131 CP1US5 136041737 IC50 = 7070 nM T94131 CXH63V 136041747 IC50 > 10000 nM T94131 C6B5TC 136041748 IC50 > 10000 nM T94131 CU6XG1 136041749 IC50 > 10000 nM T94131 C0U5DB 136041750 IC50 > 10000 nM T94131 C48KAQ 136041752 IC50 > 10000 nM T94131 C74PRL 136041753 IC50 > 10000 nM T94131 CT4FJ1 136041757 IC50 = 10000 nM T94131 CCS2G6 136041761 IC50 > 10000 nM T94131 CEZP21 136041762 IC50 > 10000 nM T94131 CJ58TD 136041764 IC50 > 10000 nM T94131 CX67QW 136041765 IC50 > 10000 nM T94131 CK0H2Q 136041766 IC50 > 10000 nM T94131 CQP7B6 136041767 IC50 > 10000 nM T94131 CM65BS 136041773 IC50 = 8270 nM T94131 C6P7JB 136041775 IC50 > 10000 nM T94131 C5CJF7 136041776 IC50 > 10000 nM T94131 C3XIZ8 136041777 IC50 > 10000 nM T94131 C32LKO 136041785 IC50 > 10000 nM T94131 C90ARP 136041787 IC50 > 10000 nM T94131 CZ3BN1 136041792 IC50 = 6215 nM T94131 CG19DI 136041799 IC50 > 10000 nM T94131 CXJA29 136041804 IC50 = 10000 nM T94131 CHT31V 136041805 IC50 = 1590 nM T94131 CO8C4J 136041817 IC50 = 3315 nM T94131 C4QU6G 136041827 IC50 = 10000 nM T94131 CNE10X 136041834 IC50 = 10000 nM T94131 CS3AE1 136041847 IC50 > 10000 nM T94131 CZC47Y 136041848 IC50 > 10000 nM T94131 C7PHA5 136044403 IC50 = 60 nM T94131 CLA3C2 136068720 IC50 = 96.5 nM T94131 CA91JG 136069599 IC50 = 1532 nM T94131 CGAB91 136069600 IC50 = 7418 nM T94131 C3ZAW2 136069605 IC50 = 8400 nM T94131 C8JXL5 136069609 IC50 = 1000 nM T94131 C9I0EQ 136069610 IC50 = 8966 nM T94131 C25EYJ 136069611 IC50 = 2461 nM T94131 C2S5QF 136069615 IC50 = 10000 nM T94131 CI1LY8 136096349 IC50 = 60 nM T94131 CC4UM3 136176116 IC50 > 10000 nM T94131 CJRK81 136176117 IC50 > 10000 nM T94131 C63IOS 136176118 IC50 > 10000 nM T94131 C3KW7H 136176119 IC50 > 10000 nM T94131 C69AKQ 136176120 IC50 > 10000 nM T94131 CF17KO 136176121 IC50 > 10000 nM T94131 CU3TE0 136176122 IC50 = 3333 nM T94131 C3X5KE 136176124 IC50 > 10000 nM T94131 CA8C5E 136176125 IC50 > 10000 nM T94131 C5OMG2 136176126 IC50 > 10000 nM T94131 CP2YM7 136176127 IC50 > 10000 nM T94131 C8XIJ0 136176128 IC50 = 5742 nM T94131 CUY8N4 136176129 IC50 > 10000 nM T94131 C3J4ME 136176130 IC50 > 10000 nM T94131 CR1NZ2 136176131 IC50 > 10000 nM T94131 C4WG2F 136176132 IC50 > 10000 nM T94131 CJ8EC5 136176139 IC50 > 10000 nM T94131 CQ84IZ 136180335 Ki > 4000 nM T94131 C1LK9U 136183381 IC50 = 3975 nM T94131 C27TKQ 136196449 IC50 = 10000 nM T94131 CHF3R5 136200721 IC50 = 4810 nM T94131 CV2X9O 136200837 IC50 = 3690 nM T94131 CK9S4X 136229137 IC50 = 18500 nM T94131 C7S1YJ 136230225 IC50 > 10000 nM T94131 C3Q6ED 136230226 IC50 > 10000 nM T94131 CKPF02 136230227 IC50 > 10000 nM T94131 CZY9O0 136230228 IC50 = 5090 nM T94131 CRET01 136230229 IC50 > 10000 nM T94131 CX1KI8 136230230 IC50 > 10000 nM T94131 C3Z5MH 136230231 IC50 > 10000 nM T94131 CUE6N8 136230232 IC50 = 8010 nM T94131 C8Q1AP 136230233 IC50 = 6710 nM T94131 C70RXE 136230234 IC50 > 10000 nM T94131 C4W0KN 136230235 IC50 = 6610 nM T94131 CMZN01 136230236 IC50 > 10000 nM T94131 CCU0H5 136241428 IC50 = 1780 nM T94131 C75RWX 136244223 IC50 = 7410 nM T94131 CXI04C 136244224 IC50 = 6480 nM T94131 C0YW6L 136244283 IC50 = 1340 nM T94131 CF3DK1 136245085 IC50 = 9360 nM T94131 CEU87Z 136245089 IC50 = 10000 nM T94131 CUF56H 136245251 IC50 = 2170 nM T94131 CKPR81 136245252 IC50 = 7120 nM T94131 C7C5ZV 136249323 IC50 = 2600 nM T94131 CI6HG4 136249373 IC50 = 264 nM T94131 CL4MO3 136249382 IC50 = 10000 nM T94131 C68CRX 136254271 IC50 = 2870 nM T94131 C0GZV9 136254283 IC50 > 10000 nM T94131 CMWA86 136264282 IC50 = 9149 nM T94131 CSD78N 136264452 IC50 = 6390 nM T94131 C1HI5T 136264454 IC50 = 1131 nM T94131 CV3UE9 137333450 IC50 = 202.7 nM T94131 CH8WU5 137348751 IC50 = 12.59 nM T94131 CP34TI 137631388 IC50 = 130 nM T94131 CF0PQ2 137632018 IC50 > 794.33 nM T94131 CZ4WN6 137633048 Ki = 66.7 nM T94131 CIX4S7 137633081 IC50 = 630.96 nM T94131 CR17XH 137634463 IC50 = 499 nM T94131 CM63EP 137634801 IC50 = 6309.57 nM T94131 CYAL31 137634808 Ki = 113 nM T94131 C34MHP 137634951 IC50 = 35 nM T94131 C9GXM1 137635017 IC50 = 794.33 nM T94131 C06BDR 137635072 IC50 = 150 nM T94131 CY86AJ 137635564 IC50 = 630.96 nM T94131 CYK6C4 137635941 IC50 >= 199.53 nM T94131 CMN6T7 137636115 IC50 = 125 nM T94131 CZ74XF 137636132 IC50 = 316.23 nM T94131 CPJ43Y 137636841 IC50 = 220 nM T94131 C7BE2O 137636964 IC50 = 10000 nM T94131 CV38QX 137637076 IC50 > 1000 nM T94131 CK4V7A 137637244 IC50 = 2511.89 nM T94131 CK2HR6 137637299 IC50 = 4300 nM T94131 CXPI97 137637422 IC50 >= 199.53 nM T94131 CX8NI0 137637899 IC50 = 15848.93 nM T94131 CMZV19 137639099 IC50 = 199.53 nM T94131 CJ3LX4 137639119 IC50 = 4.7 nM T94131 CS78JW 137639139 IC50 = 43 nM T94131 CHK7G9 137639570 IC50 = 6309.57 nM T94131 C4TSZ8 137639858 IC50 = 316.23 nM T94131 CK9GP8 137640140 Ki > 490 nM T94131 C7HA4V 137640279 IC50 >= 199.53 nM T94131 CA0QO6 137640453 IC50 = 91.9 nM T94131 CWK2F4 137640548 IC50 > 31622.78 nM T94131 C67NLM 137640896 IC50 >= 199.53 nM T94131 CQ8X0E 137641383 IC50 = 99 nM T94131 C0I6RQ 137641405 IC50 = 1000 nM T94131 CN3F5A 137641753 IC50 >= 199.53 nM T94131 C5X3TH 137642662 IC50 = 27 nM T94131 C1EBS6 137642764 Ki > 490 nM T94131 C8M9TX 137642801 IC50 = 16 nM T94131 CL4Q9G 137643238 IC50 > 1000 nM T94131 CP3JK1 137643598 IC50 = 794.33 nM T94131 CAPQ93 137644458 IC50 = 251.19 nM T94131 C4KAU7 137644907 IC50 = 7943.28 nM T94131 CKI2G8 137645541 IC50 = 398.11 nM T94131 C6SW7U 137646075 IC50 >= 199.53 nM T94131 C9SU6F 137646331 IC50 = 630.96 nM T94131 C5ERV3 137646413 IC50 = 29 nM T94131 CZC27Y 137646667 IC50 = 158.49 nM T94131 CA4V8H 137646998 IC50 >= 199.53 nM T94131 C5HIM9 137647114 IC50 = 398.11 nM T94131 CPMG65 137647250 IC50 = 8.4 nM T94131 C3TXN9 137647591 IC50 = 291 nM T94131 CPX42N 137647765 IC50 = 190 nM T94131 C6OK0J 137647964 IC50 > 19952.62 nM T94131 CS39XP 137648085 IC50 = 251.19 nM T94131 C4Z0NQ 137648826 IC50 = 1584.89 nM T94131 CE54DO 137648917 IC50 >= 199.53 nM T94131 CSML14 137649696 IC50 = 47 nM T94131 CCM18K 137650283 IC50 = 794.33 nM T94131 CHT1R8 137650579 IC50 = 794.33 nM T94131 C9QA0W 137652944 IC50 >= 199.53 nM T94131 CI64CW 137653468 IC50 > 25118.86 nM T94131 CN78RE 137653565 IC50 = 501.19 nM T94131 CTKQ38 137653713 IC50 = 199.53 nM T94131 C9M4PI 137653924 IC50 = 398.11 nM T94131 C9E5JK 137654836 IC50 = 316.23 nM T94131 CD19ZS 137654937 IC50 = 61 nM T94131 C4N5LS 137655123 IC50 = 1000 nM T94131 C82EOF 137655140 IC50 = 316.23 nM T94131 CHV26G 137655828 IC50 = 20 nM T94131 CC5NK4 137655965 IC50 = 501.19 nM T94131 CLC7N4 137656507 IC50 = 630.96 nM T94131 CE9H8D 137657006 IC50 = 1995.26 nM T94131 C3TD6A 137657429 Ki = 84.3 nM T94131 C2JX1W 137657572 IC50 >= 199.53 nM T94131 C41OPW 137658031 IC50 = 3162.28 nM T94131 C6BF8E 137658458 IC50 = 390 nM T94131 C35DPY 137658611 IC50 = 398.11 nM T94131 CU9PB7 137659393 IC50 = 501.19 nM T94131 CZ36BW 137659557 IC50 = 501.19 nM T94131 C3CF4O 137659746 IC50 = 316.23 nM T94131 CCX64Q 137660055 IC50 = 398.11 nM T94131 C1F6QN 137660818 IC50 >= 199.53 nM T94131 CP5K4E 137660883 IC50 = 132 nM T94131 C1OLQ3 137660961 IC50 = 1258.93 nM T94131 CM6FS2 137661095 IC50 = 398.11 nM T94131 C8R3JK 137661301 IC50 = 158.49 nM T94131 C9HPG8 137661516 IC50 = 1584.89 nM T94131 C90ELH 137661890 IC50 = 187 nM T94131 CA3C4O 138454792 IC50 = 67 nM T94131 CKDZ26 138504497 IC50 = 2900 nM T94131 C0BFS3 139327957 IC50 = 140 nM T94131 C7ZAQ1 141406387 IC50 = 24640 nM T94131 C7NUI8 141406388 IC50 = 42570 nM T94131 CQYI18 141406390 IC50 = 9470 nM T94131 CUA1D0 141406392 IC50 = 38290 nM T94131 CP0R6Y 141406393 IC50 = 1900 nM T94131 C1EVQ0 141406394 IC50 = 17810 nM T94131 C2QP0F 141406396 IC50 = 18240 nM T94131 CY2M0B 141406399 IC50 = 5100 nM T94131 CC3OU2 141406400 IC50 = 32180 nM T94131 CKV13Y 141406404 IC50 = 19030 nM T94131 C3Q1VL 141419885 IC50 = 174.2 nM T94131 C3EJX8 141419888 IC50 = 198.5 nM T94131 CKX4P3 141446054 IC50 > 158489.32 nM T94131 C9IV8R 141461655 IC50 = 268 nM T94131 C4C0QL 141461656 IC50 = 37 nM T94131 CG6O8P 141461658 IC50 = 63 nM T94131 C6I1VW 141461659 IC50 = 155 nM T94131 CES84U 141461662 IC50 = 1593 nM T94131 CM8HT7 141461664 IC50 = 381 nM T94131 CZV17F 141461667 IC50 = 7 nM T94131 CFR0I4 141461668 IC50 = 2062 nM T94131 CD5VE0 141461669 IC50 = 17 nM T94131 CU6LE4 141461671 IC50 = 15 nM T94131 CHJ93Y 141461672 IC50 = 2966 nM T94131 CV54CS 141471198 IC50 = 11 nM T94131 C25HYI 141471200 IC50 = 10 nM T94131 CZS03J 141509623 IC50 = 684 nM T94131 C1R9AN 141518981 IC50 = 45 nM T94131 C4MH5U 141518989 IC50 = 37 nM T94131 CQT27N 141520958 IC50 = 116 nM T94131 CH5F2X 141716982 IC50 = 1.259 nM T94131 CRU08D 141717009 IC50 = 0.7943 nM T94131 C8Q0VB 141717016 IC50 = 1.259 nM T94131 CQ34YR 142506035 IC50 = 162 nM T94131 CU03GW 142506036 IC50 = 2 nM T94131 C74MXW 142506065 IC50 = 3 nM T94131 CX6BQ7 142506102 IC50 = 2 nM T94131 CY3BM0 142506119 IC50 = 1769 nM T94131 CC6MD0 142506155 IC50 = 8 nM T94131 C05QOM 142506157 IC50 = 203 nM T94131 CGNQ74 142506189 IC50 = 103 nM T94131 CT3U9R 142506192 IC50 = 2 nM T94131 C1T3IQ 142506210 IC50 = 43 nM T94131 CEGV67 142506220 IC50 = 234 nM T94131 CP5HF8 142506225 IC50 = 995 nM T94131 C1U3CA 142506238 IC50 = 45 nM T94131 C7QMG9 145108300 IC50 = 17 nM T94131 C1FIE4 145439085 IC50 = 2293 nM T94131 CGF4I3 145946093 IC50 = 316.23 nM T94131 CI40JE 145951013 IC50 = 602.1 nM T94131 C6YT8E 145951131 IC50 > 9100 nM T94131 CFW62M 145951569 IC50 = 120.5 nM T94131 CHA84K 145951830 IC50 > 10000 nM T94131 CT4I9A 145952160 IC50 = 31 nM T94131 C91GVH 145952598 IC50 = 76 nM T94131 C1W0GJ 145952796 IC50 = 25118.86 nM T94131 CVMF13 145953272 IC50 = 1207 nM T94131 CYL5T1 145953372 IC50 <= 10000 nM T94131 CP14AV 145953653 IC50 = 751 nM T94131 CY8D5Q 145953886 IC50 = 596.3 nM T94131 C3ZUW8 145954195 IC50 = 358.3 nM T94131 C1NJB7 145955070 IC50 = 47 nM T94131 CRHE01 145955133 IC50 <= 10000 nM T94131 C7MP9Z 145955279 IC50 = 255.7 nM T94131 C7K8VT 145955565 IC50 = 118.1 nM T94131 CPU4X2 145955670 IC50 = 1898 nM T94131 C3ST5Y 145955693 IC50 = 140 nM T94131 C1VH5X 145955836 IC50 = 2628 nM T94131 C7K2YF 145956631 IC50 <= 10000 nM T94131 CQW74M 145956683 IC50 = 110 nM T94131 CJ1F6A 145956725 IC50 = 1036 nM T94131 C12IFO 145956886 IC50 = 456.7 nM T94131 C9O2PL 145958063 IC50 = 193.7 nM T94131 CQH01X 145958257 IC50 <= 10000 nM T94131 C3DGU7 145958571 IC50 = 708 nM T94131 C9NS6T 145958690 IC50 = 245.5 nM T94131 C7ZO9V 145959196 IC50 = 236 nM T94131 CSC81H 145959429 IC50 = 62 nM T94131 C0S1YM 145959980 IC50 = 303 nM T94131 CT3I2R 145960112 IC50 = 893.1 nM T94131 C8MJ9X 145960272 IC50 = 170 nM T94131 CLH5J2 145960703 IC50 = 6.31 nM T94131 CF36RA 145961004 IC50 = 64 nM T94131 CZO6T7 145961089 IC50 = 2511.89 nM T94131 CX6T3J 145961172 IC50 > 10000 nM T94131 C9I7EC 145961182 IC50 = 7.943 nM T94131 C54ZQA 145961234 IC50 = 3981.07 nM T94131 C83FPK 145961240 IC50 = 100 nM T94131 C31QBE 145961348 IC50 > 10000 nM T94131 CHF56O 145961403 IC50 > 9100 nM T94131 C2GT9Y 145961404 IC50 > 9100 nM T94131 COCG81 145961565 IC50 = 6309.57 nM T94131 C73MVW 145961583 IC50 = 1584.89 nM T94131 CKF0I1 145961740 IC50 = 1.259 nM T94131 C6HB9M 145961899 IC50 = 6309.57 nM T94131 CS46RM 145962397 Ki = 160 nM T94131 CT42OW 145962848 IC50 = 25.12 nM T94131 CLFQ85 145963006 IC50 = 12.59 nM T94131 CAI0D6 145963117 IC50 = 256 nM T94131 CA4FO3 145963201 IC50 = 10 nM T94131 CYZ14S 145963250 IC50 = 7943.28 nM T94131 CAD5Q9 145963302 IC50 > 10000 nM T94131 C35ZRP 145963416 IC50 > 10000 nM T94131 CQBU31 145963478 IC50 > 1000 nM T94131 C0S1ZI 145963484 IC50 = 1.259 nM T94131 C4JI8B 145963558 IC50 = 158.49 nM T94131 C87HFG 145964719 IC50 = 4752 nM T94131 CRE3Q1 145966313 IC50 = 68 nM T94131 CU9XC4 145966764 IC50 = 0.7 nM T94131 C97IKW 145969580 IC50 = 223.9 nM T94131 CK82QG 145969816 IC50 = 1783 nM T94131 C71YAK 145970017 IC50 = 3000 nM T94131 C3Y7RS 145970202 IC50 > 10000 nM T94131 CP6YC2 145970436 IC50 = 117.5 nM T94131 CZ98FH 145971490 IC50 = 1591 nM T94131 CTB97Z 145971948 IC50 = 408 nM T94131 CGQJ04 145972017 IC50 = 1590 nM T94131 C96IUM 145973569 IC50 = 0.5 nM T94131 CD7PS3 145973794 IC50 = 420 nM T94131 CZ9G6E 145974533 IC50 = 146 nM T94131 C3XIT8 145974725 IC50 = 1491 nM T94131 C1N5TZ 145975623 IC50 = 445 nM T94131 C3LR4O 145976442 IC50 = 3560 nM T94131 C3YG4Z 145977475 IC50 = 0.7 nM T94131 CPZS56 145982349 EC50 = 10000 nM T94131 CH90CT 145983168 IC50 = 184.7 nM T94131 CJU02I 145983624 IC50 = 62 nM T94131 CVS2U0 145983808 IC50 = 363 nM T94131 CF8MR5 145986347 IC50 = 1000 nM T94131 C6XMQ8 145989163 EC50 = 9890 nM T94131 CBU86Y 145991850 IC50 = 10000 nM T94131 C8X2IT 145996536 IC50 > 10000 nM T94131 C4K0JW 145996540 IC50 = 1.2 nM T94131 C6RPG0 146014481 IC50 = 831.76 nM T94131 C59KOM 146585662 IC50 = 9 nM T94131 CFQO97 146585699 IC50 = 752 nM T94131 C0GMR1 146585718 IC50 = 135 nM T94131 CI85VS 146731761 IC50 = 81 nM T94131 CWZ05D 148564044 IC50 = 22 nM T94131 C4MC0S 149169124 IC50 = 1870 nM T94131 CVW62P 149242889 IC50 = 10530 nM T94131 CN87RZ 149370890 IC50 = 810 nM T94131 CK4FJ1 149556361 IC50 = 2300 nM T94131 C8UQL4 153940691 IC50 = 1320 nM T94131 CMZ68Q 153940692 IC50 = 110 nM T94131 C5X7JK 154734328 IC50 = 1000 nM T94131 C8Q9UG 155510876 IC50 = 222 nM T94131 CDT8F2 155510913 IC50 = 1258.93 nM T94131 C6WIC9 155511977 IC50 = 1258.93 nM T94131 CPH8N1 155512095 IC50 = 251.19 nM T94131 CZJ9D6 155512258 IC50 = 5533 nM T94131 CG9I4X 155512515 IC50 = 140 nM T94131 CR1Z8A 155512529 IC50 > 10000 nM T94131 CQZY50 155512775 IC50 = 39.81 nM T94131 C5V2GO 155512947 IC50 = 2511.89 nM T94131 C1DIT4 155513047 IC50 = 125.89 nM T94131 C8PG6Z 155513084 IC50 = 794.33 nM T94131 C5M6NS 155513226 IC50 = 9550 nM T94131 C45SYX 155513615 IC50 = 6 nM T94131 CBH57O 155514764 IC50 = 2511.89 nM T94131 C5C9EG 155515047 IC50 = 1000 nM T94131 CEFS61 155515135 IC50 = 2650 nM T94131 C0AXF7 155515394 IC50 = 1584.89 nM T94131 CTS48F 155515676 IC50 = 3 nM T94131 C7Q3FR 155515734 IC50 = 1995.26 nM T94131 C30ZFN 155516445 IC50 = 630.96 nM T94131 CJDG04 155516604 IC50 = 100 nM T94131 C42JXQ 155517064 IC50 = 1995.26 nM T94131 CYO19V 155517071 IC50 = 125.89 nM T94131 CYWX76 155517213 IC50 = 1584.89 nM T94131 CT53XD 155517442 IC50 = 12589.25 nM T94131 C4G8YN 155517534 IC50 = 1983 nM T94131 CS2JT9 155518175 IC50 = 3162.28 nM T94131 CW7OM6 155518918 IC50 = 708 nM T94131 CC51GM 155519635 IC50 = 158.49 nM T94131 CHFJ25 155519726 IC50 = 12589.25 nM T94131 CZ78HW 155519830 IC50 = 316.23 nM T94131 CQEK39 155520373 IC50 = 4.3 nM T94131 C3D7FJ 155520444 IC50 = 6309.57 nM T94131 C5D6YX 155521099 IC50 > 10000 nM T94131 CEA3M1 155521494 IC50 = 63.1 nM T94131 CBSR95 155522042 IC50 = 3480 nM T94131 CZO7Q8 155522149 IC50 = 536 nM T94131 CCGW06 155523124 IC50 = 6309.57 nM T94131 CNB70P 155523246 IC50 = 1000 nM T94131 C4TLQ7 155523447 IC50 > 10000 nM T94131 CZG27I 155523570 IC50 = 38 nM T94131 C37RVF 155523599 IC50 = 4500 nM T94131 C4H2AB 155524238 IC50 = 15.85 nM T94131 CP18VT 155524467 IC50 = 1995.26 nM T94131 CUP7L2 155524901 IC50 = 1258.93 nM T94131 C2BL5I 155525312 IC50 = 25.12 nM T94131 C10RZQ 155525477 IC50 = 1000 nM T94131 CF76OV 155525717 IC50 = 19.3 nM T94131 C0UA4D 155525996 IC50 = 63.1 nM T94131 C0AR4W 155526097 IC50 = 3981.07 nM T94131 C3EAR8 155526323 IC50 = 1000 nM T94131 C82NUW 155527501 IC50 = 445 nM T94131 CK07GS 155527559 IC50 = 64 nM T94131 CX12MK 155527651 IC50 = 4 nM T94131 C8Z3TK 155528581 IC50 = 1584.89 nM T94131 C0B2NV 155528644 IC50 = 853 nM T94131 C3VAI9 155528997 IC50 = 501.19 nM T94131 C9L6OC 155529247 IC50 = 467 nM T94131 C2FE1S 155529479 IC50 = 25.12 nM T94131 CB90AR 155529643 IC50 = 199.53 nM T94131 CFV1S0 155529706 IC50 = 434 nM T94131 C14QOF 155530163 IC50 = 1584.89 nM T94131 C4I5UP 155530224 IC50 = 158.49 nM T94131 CX6N3Y 155531155 IC50 = 79.43 nM T94131 C9AXO7 155531257 IC50 = 1258.93 nM T94131 CGAI60 155531409 IC50 = 3162.28 nM T94131 CDI4V8 155531526 IC50 = 194 nM T94131 CE6QP1 155532037 IC50 = 501.19 nM T94131 CJH9U4 155532237 IC50 = 12589.25 nM T94131 C6W0JX 155532471 IC50 = 6309.57 nM T94131 CKMD29 155532546 IC50 = 6309.57 nM T94131 C3XFB8 155532820 IC50 = 19.95 nM T94131 CIYA39 155532858 IC50 = 34 nM T94131 C0GR1J 155533050 IC50 = 2 nM T94131 CQS8P1 155533070 IC50 = 1584.89 nM T94131 C0SZR9 155533335 IC50 = 2511.89 nM T94131 CAT9V1 155533370 IC50 = 5600 nM T94131 C67ERP 155533384 IC50 = 158.49 nM T94131 CL8OM7 155533564 IC50 = 6081 nM T94131 CBM24U 155533579 IC50 = 3981.07 nM T94131 CR5H8B 155533591 IC50 = 1995.26 nM T94131 CA7T0Y 155533911 IC50 = 9340 nM T94131 C8XQ4W 155534168 IC50 = 87 nM T94131 CN1ST4 155534269 IC50 = 1258.93 nM T94131 CBEG39 155534594 IC50 = 1258.93 nM T94131 CTZ3E0 155534905 IC50 = 112 nM T94131 CG1JR7 155535513 IC50 = 630.96 nM T94131 CN6KJ5 155535520 IC50 = 794.33 nM T94131 C5F2TY 155535537 IC50 = 1995.26 nM T94131 CKB2U4 155535691 IC50 = 63.1 nM T94131 CY7X3M 155535740 IC50 = 39.81 nM T94131 CUWE49 155535963 IC50 = 794.33 nM T94131 C70UDF 155536179 IC50 = 3162.28 nM T94131 CEJ6L1 155536226 IC50 = 210.7 nM T94131 CNB24M 155536473 IC50 = 1000 nM T94131 C2CG1A 155537016 IC50 = 3981.07 nM T94131 C8AJ6C 155538256 IC50 = 250.4 nM T94131 CQ1E6H 155538266 IC50 = 39.81 nM T94131 CZ19AN 155538609 IC50 = 496 nM T94131 CHR8M1 155538990 IC50 = 7510 nM T94131 CC1BG2 155539321 IC50 > 10000 nM T94131 CF20PS 155539394 IC50 = 2511.89 nM T94131 C8LKW4 155540264 IC50 = 2511.89 nM T94131 C6I5DK 155541290 IC50 = 1258.93 nM T94131 CECX47 155541544 IC50 = 501.19 nM T94131 C4FC0V 155541900 IC50 = 630.96 nM T94131 CKBW37 155542030 IC50 = 1905 nM T94131 CASE16 155542363 IC50 = 3162.28 nM T94131 C8AXF9 155542633 IC50 = 5011.87 nM T94131 C8OC2P 155542800 IC50 = 5600 nM T94131 C42BIZ 155542813 IC50 = 12589.25 nM T94131 CVNR95 155542898 IC50 = 1400 nM T94131 C1SY0G 155543154 IC50 = 23200 nM T94131 C7IWJ2 155543389 IC50 = 10000 nM T94131 CZY0N4 155543588 IC50 = 10 nM T94131 CJB8C9 155543659 IC50 = 231 nM T94131 CX1C8I 155544561 IC50 > 10000 nM T94131 CBN29V 155544583 IC50 = 204 nM T94131 C98FXC 155544955 IC50 = 3594 nM T94131 CTSW53 155546042 IC50 > 10000 nM T94131 CQ6J7U 155546361 IC50 = 280 nM T94131 C8SQA2 155546999 IC50 = 12.59 nM T94131 C8D4ZH 155547166 IC50 = 630.96 nM T94131 CI6KO7 155548518 IC50 = 251.19 nM T94131 CL4F8P 155549003 IC50 = 7.943 nM T94131 CM6S8K 155549098 IC50 = 5011.87 nM T94131 C4PEJ5 155549895 IC50 > 10000 nM T94131 CFP94J 155550309 IC50 = 794.33 nM T94131 CQ5OD0 155550395 IC50 = 45 nM T94131 CK1JR7 155551961 IC50 = 6.5 nM T94131 CJ75BO 155552100 IC50 > 1000 nM T94131 CXN3Y8 155553327 IC50 = 3981.07 nM T94131 CL04BD 155554125 IC50 = 934 nM T94131 CX9C6O 155554180 IC50 = 1000 nM T94131 CC13QL 155555170 IC50 = 1378 nM T94131 CZX06J 155555458 IC50 = 1995.26 nM T94131 C2OGW1 155555483 IC50 = 521 nM T94131 CRO5Z3 155556073 IC50 = 5756 nM T94131 CH2P4T 155556124 IC50 = 25118.86 nM T94131 CCU8M1 155556480 IC50 = 15848.93 nM T94131 CIU29Z 155556576 IC50 > 10000 nM T94131 CM3LI6 155556593 IC50 > 10000 nM T94131 CZ8CX1 155556887 IC50 = 501.19 nM T94131 CG2FS6 155557123 IC50 = 2511.89 nM T94131 CFS63H 155557182 IC50 = 301 nM T94131 C0FE4G 155557988 IC50 = 2183 nM T94131 CR8J0E 155558167 IC50 = 50.12 nM T94131 CN96JH 155558197 IC50 = 316.23 nM T94131 CSO4M3 155558261 IC50 = 5011.87 nM T94131 C52TSP 155558262 IC50 = 440 nM T94131 CS70ER 155559192 IC50 = 247 nM T94131 CVG49I 155560688 IC50 = 4010 nM T94131 C5S7AL 155560766 IC50 = 199.53 nM T94131 CQ7PS9 155560780 IC50 = 3981.07 nM T94131 CLO3B1 155561152 IC50 = 7900 nM T94131 C8XS0L 155561165 IC50 = 794.33 nM T94131 C72CQG 155561233 IC50 = 125.89 nM T94131 C1INL7 155561328 IC50 = 794.33 nM T94131 CX6U2T 155562388 IC50 = 3981.07 nM T94131 C5E9TP 155562641 IC50 = 79432.82 nM T94131 CCF4W2 155563986 IC50 = 6309.57 nM T94131 CHK4E8 155565269 IC50 = 1258.93 nM T94131 C7PXA0 155565551 IC50 = 630.96 nM T94131 CY4N7O 155565715 IC50 = 15848.93 nM T94131 CVQ6Z4 155565763 IC50 = 2511.89 nM T94131 CA1RX3 155565771 IC50 = 2511.89 nM T94131 CQ3AU4 155565828 IC50 = 19952.62 nM T94131 CMK4I3 155565845 IC50 = 1995.26 nM T94131 C59VPW 155565958 IC50 = 1584.89 nM T94131 CAP9F2 155566187 IC50 = 15 nM T94131 CM7E2G 155566279 IC50 = 3162.28 nM T94131 C3BNY5 155566309 IC50 = 10000 nM T94131 C9KQW3 155567372 IC50 = 740 nM T94131 C98NZE 155567616 IC50 = 5011.87 nM T94131 C1HQ5J 155568324 IC50 = 354 nM T94131 CLA46O 155568356 IC50 = 800 nM T94131 C7SLR8 155568452 IC50 = 501.19 nM T94131 C1S8ZB 155568922 IC50 > 1000 nM T94131 C14LVO 155569074 IC50 = 158.49 nM T94131 CFWP17 155569113 IC50 = 587 nM T94131 CUH38L 155569363 IC50 = 8420 nM T94131 C4H0NE 155569598 IC50 = 3162.28 nM T94131 D00GQM 25069592 IC50 = 7972 nM T94131 D00ZIK 9908783 IC50 = 61000 nM T94131 D01ILN 223355 IC50 = 8500 nM T94131 D01SSI 24937012 IC50 > 10000 nM T94131 D03EHM 24905142 IC50 = 1100 nM T94131 D03QQH 16760391 IC50 = 100000 nM T94131 D05USL 5278396 IC50 > 1000 nM T94131 D06DNH 9907093 IC50 > 10000 nM T94131 D06HVH 54613583 IC50 = 3100 nM T94131 D06PWI 42623951 IC50 = 25.12 nM T94131 D07JKB 135955185 IC50 = 5135 nM T94131 D07PMP 44187953 IC50 = 16 nM T94131 D08KSQ 11637090 IC50 > 10000 nM T94131 D08NQM 5289247 IC50 = 8 nM T94131 D09FBN 135955186 IC50 = 8558 nM T94131 D09ZNV 447682 IC50 > 200000 nM T94131 D0AH8Q 25074311 IC50 = 6742 nM T94131 D0EU1R 46215815 IC50 = 25118 nM T94131 D0F1SI 25074312 IC50 = 8000 nM T94131 D0H0HR 49836027 IC50 = 171 nM T94131 D0H2CM 135565635 IC50 = 1300 nM T94131 D0P5TI 58441401 IC50 = 240.3 nM T94131 D0R0TW 11964036 IC50 = 590 nM T94131 D0R2UG 52936849 IC50 = 104 nM T94131 D0S5YV 6852167 Ki = 7 nM T94131 D0T3PW 5281672 IC50 = 4720 nM T94131 D0TC5H 16049458 IC50 = 2343 nM T94131 D0W8XH 9884685 IC50 = 15 nM T94131 D0Y1DR 46225260 IC50 = 7371 nM T94131 D0Y3OO 11327430 IC50 = 220 nM T16042 D02HWP 2722 IC50 = 2400 nM T16042 D04AIT 5280445 IC50 = 5000 nM T16042 D09JUG 60490 IC50 = 400 nM T16042 D0H2DQ 4912 IC50 = 14000 nM T16042 D0K8KX 5280343 IC50 = 2200 nM T16042 D0DK4I 4534 IC50 = 4900 nM T16042 D0DP8P 47795 IC50 = 213000 nM T16042 D0J8RS 297589 IC50 = 810 nM T16042 CD6W3K 6618 IC50 = 4000 nM T16042 CUO98K 7808 IC50 = 55000 nM T16042 C6Q1HE 9230 Ki = 25000 nM T16042 CFQ35W 11563 IC50 > 100000 nM T16042 C4T5QC 11847 IC50 > 100000 nM T16042 C0NHG2 12005 IC50 = 34000 nM T16042 CP1V2F 68523 IC50 > 100000 nM T16042 C9CLG6 70119 IC50 > 100000 nM T16042 CQ1G7S 70840 IC50 > 50000 nM T16042 CY0AL9 72279 IC50 > 100000 nM T16042 C6CLP5 80801 IC50 = 5000 nM T16042 C0JLT2 125100 IC50 > 100000 nM T16042 CDV60U 125101 IC50 = 510 nM T16042 CUP4Y3 128132 IC50 = 40000 nM T16042 C1H8NR 155248 IC50 = 1210 nM T16042 CDN7P9 156398 IC50 = 150 nM T16042 C7FL5H 173513 IC50 = 19000 nM T16042 CAL71Q 255670 IC50 > 100000 nM T16042 C0SMD7 339231 IC50 = 790 nM T16042 C05QAO 353995 IC50 > 100000 nM T16042 C9XA6R 356358 IC50 = 5700 nM T16042 CF2YR7 356359 IC50 = 3700 nM T16042 CS0DT8 476858 IC50 = 580 nM T16042 CVJ0B7 614686 IC50 = 7000 nM T16042 C97DNA 637177 IC50 = 59000 nM T16042 CA9BW2 637234 IC50 = 1000 nM T16042 CGT7F0 661037 IC50 = 25000 nM T16042 CVN7D4 663428 IC50 = 100 nM T16042 CV97HM 663693 Ki = 19 nM T16042 CWB50H 663890 IC50 = 3000 nM T16042 CS8OW2 663999 IC50 > 40000 nM T16042 CZ4O7G 664510 Ki = 100 nM T16042 CSJ9X8 668390 IC50 = 618 nM T16042 C2WLD1 685709 IC50 > 50000 nM T16042 CJ2L1C 688659 IC50 > 100000 nM T16042 C2XMJ8 693672 IC50 = 15000 nM T16042 C04WFD 697726 IC50 = 6000 nM T16042 C2SG4A 698916 IC50 = 17000 nM T16042 CCY5N0 727302 IC50 > 100000 nM T16042 CF9HW0 754454 IC50 = 292 nM T16042 CBM8Y0 771546 IC50 > 100000 nM T16042 C3ZD2R 775981 IC50 = 7000 nM T16042 C17CVK 775988 IC50 = 10000 nM T16042 CJ1U3G 775990 IC50 > 50000 nM T16042 CPM12N 775994 IC50 = 3400 nM T16042 CWER09 775998 IC50 = 18000 nM T16042 CMY7U5 776006 IC50 = 10000 nM T16042 CMA8X3 776051 IC50 = 9100 nM T16042 CA2VY1 776057 IC50 = 7000 nM T16042 C9Z8TL 781202 IC50 = 20000 nM T16042 C5PA3G 781212 IC50 = 4000 nM T16042 C69NGK 781217 IC50 = 11000 nM T16042 CF3KT2 781225 IC50 = 11000 nM T16042 C2VPH3 781243 IC50 = 6600 nM T16042 CIHN92 785627 IC50 = 18800 nM T16042 C0BD2V 801015 IC50 > 200000 nM T16042 C64NSF 819511 IC50 > 50000 nM T16042 CVF50J 836505 IC50 > 50000 nM T16042 CN2BT6 838850 IC50 > 50000 nM T16042 CF2MW6 854652 IC50 = 9200 nM T16042 CS26WL 874817 IC50 > 50000 nM T16042 C9QO5R 883201 IC50 > 50000 nM T16042 COE63U 889785 IC50 > 50000 nM T16042 C3ZI5M 921980 IC50 > 50000 nM T16042 CH96BV 936906 IC50 > 50000 nM T16042 CCYS81 974197 IC50 = 120 nM T16042 CIEY41 1072992 IC50 > 50000 nM T16042 CA1TU5 1079729 IC50 > 50000 nM T16042 CFO62A 1082938 IC50 > 100000 nM T16042 CG6KC7 1095055 IC50 > 100000 nM T16042 C81MSC 1141363 IC50 > 50000 nM T16042 CWE1Y9 1304061 IC50 > 100000 nM T16042 CUD6L7 1325172 IC50 > 100000 nM T16042 CW1JO4 1346428 IC50 > 100000 nM T16042 C72CAB 1550607 IC50 = 23900 nM T16042 C8Z2PM 1743704 IC50 > 100000 nM T16042 C2ROK0 1781413 IC50 = 16700 nM T16042 C1FVO5 1858274 IC50 > 50000 nM T16042 CCG73Q 1871033 Ki = 26 nM T16042 CHP4C8 1943830 Ki = 31 nM T16042 CC25XB 1998811 Ki < 10 nM T16042 C4DBG2 1998940 Ki < 10 nM T16042 CMBK51 1999882 Ki < 10 nM T16042 CQ7G5L 2013455 Ki < 10 nM T16042 CAS0O4 2013647 Ki = 170 nM T16042 C4QL9B 2017368 Ki = 15 nM T16042 CAJ10O 2192753 IC50 > 100000 nM T16042 CD0X5M 2920571 IC50 > 50000 nM T16042 CU16KY 2920793 IC50 > 25000 nM T16042 C4UJQ1 2921716 IC50 > 25000 nM T16042 C92GBS 2931181 IC50 > 100000 nM T16042 CZ02OG 2933060 IC50 > 100000 nM T16042 C1OTU9 3136123 IC50 > 50000 nM T16042 C3G9QL 3136134 IC50 > 50000 nM T16042 C35HXD 3152427 Ki = 3500 nM T16042 CPEZ98 3750129 IC50 = 10000 nM T16042 C6YJB1 4591751 IC50 = 3000 nM T16042 CV3O8W 4675130 Ki < 10 nM T16042 CF3NM8 5280701 IC50 > 25000 nM T16042 C17CBF 5281812 IC50 > 100000 nM T16042 C2NKF5 5283162 IC50 = 3000 nM T16042 C0WXP5 5284649 IC50 = 49000 nM T16042 C6IVR9 5317326 IC50 = 250 nM T16042 C6D3GZ 5393151 IC50 = 3300 nM T16042 CV56UY 5407860 IC50 = 13000 nM T16042 CV0B7K 5481241 IC50 = 7800 nM T16042 C7P4ZA 5713107 IC50 > 100000 nM T16042 CQZ8U3 6446027 IC50 > 100000 nM T16042 CTV92K 7015027 IC50 = 2000 nM T16042 CS4MF3 9586795 IC50 = 6800 nM T16042 C4T9ES 10020717 IC50 = 300 nM T16042 C1TAC5 10042678 IC50 = 24200 nM T16042 CQG4A3 10045891 IC50 = 1470 nM T16042 C20LUF 10072931 IC50 = 83 nM T16042 CKDW09 10283379 IC50 = 12000 nM T16042 CI4VW1 10316643 IC50 = 300 nM T16042 CF8Y2Q 10340455 IC50 = 350 nM T16042 CZ8B7D 10348509 IC50 = 2200 nM T16042 C3U5BM 10384947 IC50 = 300 nM T16042 C4NXL5 10554258 IC50 = 10000 nM T16042 CV0RN7 10905139 IC50 = 380 nM T16042 C13UBC 10914853 IC50 = 1000 nM T16042 C0OX8Y 10936155 IC50 = 8300 nM T16042 CWN43C 10937563 IC50 = 65 nM T16042 C1R5SB 10955008 IC50 > 100000 nM T16042 CHT16X 11019578 IC50 > 10000 nM T16042 C9IH6W 11041857 IC50 > 100000 nM T16042 C7IGY5 11142891 IC50 = 160 nM T16042 CA4TQ6 11248759 Ki = 21 nM T16042 CDL0Z1 11552655 IC50 = 85 nM T16042 C9A5QB 11741221 IC50 = 1670 nM T16042 CD3I5T 12066244 IC50 > 100000 nM T16042 CT02RU 12109338 IC50 = 42600 nM T16042 C7Y1XF 14852609 IC50 = 3900 nM T16042 C6GVK4 14983007 IC50 > 100000 nM T16042 C1YO9X 15135539 IC50 = 7300 nM T16042 C37GWC 15411433 IC50 = 39500 nM T16042 CNHZ34 15628203 IC50 = 210 nM T16042 C82ACD 16659607 IC50 = 42 nM T16042 C1JYR3 16659761 IC50 = 112 nM T16042 CCV42S 16659767 IC50 = 37 nM T16042 CK04TJ 16659930 IC50 = 117 nM T16042 C5ZM1D 16659933 IC50 = 279 nM T16042 CXL4Q3 16663122 IC50 = 99 nM T16042 C10DHE 16667292 IC50 = 26 nM T16042 C5IXG0 18822680 IC50 = 6300 nM T16042 C9WDR1 21270142 IC50 = 6200 nM T16042 CBJ87P 21270161 IC50 = 11000 nM T16042 CT94AD 21270186 IC50 = 350 nM T16042 CXQW24 21831939 IC50 > 100000 nM T16042 CS80UM 23043596 IC50 = 400 nM T16042 CQD7W3 23043614 IC50 = 5000 nM T16042 C78UAG 23043622 IC50 = 400 nM T16042 CGVH48 23043630 IC50 > 25000 nM T16042 CEFB61 23093378 IC50 > 100000 nM T16042 CBV19H 23425708 IC50 > 200000 nM T16042 CJ1O8K 23656213 IC50 = 38600 nM T16042 C4YJM0 24721289 IC50 > 100000 nM T16042 CK1SG7 24825377 Ki = 73 nM T16042 CBY15M 33845371 IC50 = 9000 nM T16042 CR74ZY 44142073 IC50 = 10000 nM T16042 CP63YR 44142076 IC50 = 25000 nM T16042 C90EVJ 44142082 Ki = 15 nM T16042 C9QXD0 44142083 Ki = 470 nM T16042 C1Q4OM 44142084 Ki = 22 nM T16042 C5MH3S 44142085 Ki = 870 nM T16042 C70VKE 44142086 Ki = 76 nM T16042 CVDX35 44246516 Ki = 2000 nM T16042 CC85WT 44318018 IC50 = 1950 nM T16042 C74QZP 44318019 IC50 = 1010 nM T16042 C4TS9J 44318030 IC50 = 1270 nM T16042 C37APD 44323089 IC50 = 85 nM T16042 C0CZ6I 44384554 IC50 = 400 nM T16042 C0Z7KU 44384614 IC50 = 1500 nM T16042 C8RZW0 44384827 IC50 > 25000 nM T16042 C3VU9Z 44385224 IC50 > 25000 nM T16042 C8QB5A 44385225 IC50 = 5000 nM T16042 C37PTI 44385415 IC50 = 600 nM T16042 CJW8D9 44385457 IC50 > 25000 nM T16042 CVPF53 44385459 IC50 = 1200 nM T16042 CGIL38 44385537 IC50 > 25000 nM T16042 CZAF84 44386778 IC50 = 28800 nM T16042 C0BRV6 44396187 IC50 = 110 nM T16042 C1TG8O 44421367 IC50 = 17000 nM T16042 CXWZ08 44421374 IC50 = 10000 nM T16042 CW8GB6 44421383 IC50 > 125000 nM T16042 COH1B3 44436892 IC50 = 7600 nM T16042 CXF24P 44437715 IC50 > 100000 nM T16042 CI7NA6 44437716 IC50 > 100000 nM T16042 C8GU3K 44437717 IC50 = 38000 nM T16042 C5I9VM 44437718 IC50 > 100000 nM T16042 C3VE4H 44437719 IC50 > 100000 nM T16042 CXK29W 44437720 IC50 > 100000 nM T16042 C9B0CX 44437721 IC50 > 100000 nM T16042 CV6W4R 44437722 IC50 > 100000 nM T16042 C7RWS3 44437723 IC50 = 18000 nM T16042 CN40UP 44437724 IC50 > 100000 nM T16042 CVBQ79 44437725 IC50 > 100000 nM T16042 C40KOY 44437726 IC50 > 100000 nM T16042 CJ1DA0 44437727 IC50 > 100000 nM T16042 C4KD8Z 44437728 IC50 > 100000 nM T16042 CWMX75 44437729 IC50 > 100000 nM T16042 C2WSB6 44437731 IC50 > 100000 nM T16042 CQT74A 44437732 IC50 = 210 nM T16042 C3M0KB 44440174 IC50 = 21600 nM T16042 C74DFE 44440176 IC50 = 9400 nM T16042 CU8L9H 44440177 IC50 = 15000 nM T16042 C3SRV6 44440179 IC50 = 33600 nM T16042 C4J6AM 44440180 IC50 = 15000 nM T16042 CDTH69 44460106 Ki = 1300 nM T16042 COD5F2 44460109 Ki < 10 nM T16042 C3B1YD 44460110 Ki < 10 nM T16042 CBOF34 44460111 Ki < 10 nM T16042 C2XZV9 44460112 Ki < 10 nM T16042 CW5Q0I 44460113 Ki = 16 nM T16042 CNK7B4 44460114 Ki < 10 nM T16042 CA7U3R 44460115 Ki < 10 nM T16042 CC86TD 44460116 Ki < 10 nM T16042 CA03BM 44460117 Ki = 33 nM T16042 CMWK84 44460120 Ki < 10 nM T16042 C9XQK7 44460121 Ki < 10 nM T16042 CG1I0J 44460122 Ki < 10 nM T16042 C7W1HI 44460123 Ki < 10 nM T16042 C9PM0I 44460124 Ki = 100 nM T16042 C0OHT1 44460125 Ki = 270 nM T16042 C3N1FC 44460126 Ki = 85 nM T16042 C37QBL 44460127 Ki < 10 nM T16042 C4B0ZM 44460128 Ki < 10 nM T16042 C8L0ZV 44460129 Ki = 27 nM T16042 C9OR2U 44460130 Ki < 10 nM T16042 CZI7W9 44460132 Ki = 1000 nM T16042 C7HIS1 44460133 Ki = 82 nM T16042 C1K4SJ 44460134 Ki = 43 nM T16042 CP1S7N 44460135 Ki = 57 nM T16042 CJM15L 44460136 Ki = 81 nM T16042 C2RU6H 44460137 Ki < 10 nM T16042 CV5BO8 44460138 Ki < 10 nM T16042 CX4GJ6 44460139 Ki < 10 nM T16042 CS29LD 44460141 Ki = 140 nM T16042 C2XWI4 44460175 IC50 > 30000 nM T16042 C85LQH 44460420 IC50 = 1450 nM T16042 CMZ5E8 44460480 IC50 = 1510 nM T16042 C0QD8O 44557858 IC50 > 150000 nM T16042 CJX28F 46213934 IC50 > 10000 nM T16042 CVW37Q 46841209 IC50 = 6800 nM T16042 CNH8K4 46841210 IC50 > 100000 nM T16042 C82JBH 46905978 IC50 = 15000 nM T16042 C2PL3G 46927848 IC50 > 10000 nM T16042 C96BOE 47168936 IC50 = 9820 nM T16042 CA4N3P 47168962 IC50 = 4090 nM T16042 CFH8P0 47169026 IC50 = 10940 nM T16042 CVMD46 47169041 IC50 = 13020 nM T16042 CCA1S4 47169049 IC50 > 20000 nM T16042 CDI71G 47172452 IC50 = 6880 nM T16042 CB8IU2 47172537 IC50 = 9380 nM T16042 C89MXP 49787910 Ki = 600 nM T16042 C4NA6U 49787911 Ki > 70000 nM T16042 C2UJF6 49787985 Ki = 26 nM T16042 CMQ45Y 49787986 Ki > 100000 nM T16042 CN4C8A 49788565 Ki < 10 nM T16042 CB7XA0 49788946 Ki < 10 nM T16042 C4O0QK 49821278 IC50 > 20000 nM T16042 CT1XC4 49852806 IC50 = 300 nM T16042 CWC6K4 49853061 IC50 > 30000 nM T16042 CC87NF 49853164 IC50 > 50000 nM T16042 C64KTI 51042131 IC50 > 10000 nM T16042 CBA28F 53299922 IC50 = 12800 nM T16042 C8G2OI 53301731 IC50 > 100000 nM T16042 CUO4X5 53301733 IC50 > 100000 nM T16042 CPNL52 53358322 IC50 = 51 nM T16042 C12BDW 53383638 Ki = 3300 nM T16042 CX4I1O 53383641 IC50 = 29800 nM T16042 CZ2WO5 53383646 IC50 = 18600 nM T16042 C2EQ8I 53383650 IC50 = 20600 nM T16042 CY9IZ6 53383655 IC50 = 24600 nM T16042 CP4LF8 53484007 IC50 > 50000 nM T16042 C5GRB6 54754354 IC50 > 10000 nM T16042 C3YM2E 54754518 IC50 > 10000 nM T16042 C5OCM9 56588198 IC50 > 100000 nM T16042 C39QPM 56588229 IC50 > 100000 nM T16042 C7ZI3H 56642018 IC50 > 10000 nM T16042 CU1G5A 56642290 IC50 > 10000 nM T16042 C0SM7Z 56642536 IC50 > 10000 nM T16042 C6TLW3 56642537 IC50 > 10000 nM T16042 CH4V1T 58567931 Ki = 250 nM T16042 C8YR9B 62197753 IC50 > 40000 nM T16042 C6DQ2M 63549790 IC50 > 40000 nM T16042 C5G0XT 65644005 IC50 > 40000 nM T16042 CJ48CY 66939548 IC50 = 1207 nM T16042 CV4P8X 68436207 IC50 = 130 nM T16042 CT70VO 68436927 IC50 = 141 nM T16042 CAD54H 70679557 IC50 > 100000 nM T16042 CPB87A 70682764 IC50 = 15600 nM T16042 CVC7A9 70691185 IC50 = 1300 nM T16042 CC03SY 70693289 IC50 = 3600 nM T16042 CC4L9K 70697403 IC50 = 12800 nM T16042 C4GE5W 70697404 IC50 > 50000 nM T16042 CA76MQ 70701378 IC50 > 70000 nM T16042 C92ZAQ 70701385 IC50 = 690 nM T16042 CRJ4S1 70701387 IC50 = 7600 nM T16042 CK3O6T 70701411 IC50 = 1300 nM T16042 CGWB74 70701426 IC50 = 9700 nM T16042 CT4IL7 70701432 IC50 > 100000 nM T16042 CK42AJ 70701448 IC50 = 730 nM T16042 C62HDV 70701451 IC50 > 40000 nM T16042 CR9AD7 70701452 IC50 > 40000 nM T16042 CD2R3J 70701454 IC50 > 40000 nM T16042 CT3SC9 70701455 IC50 > 30000 nM T16042 C30AUK 70701456 IC50 > 30000 nM T16042 CP2K1E 70701458 IC50 = 3900 nM T16042 C7QGY0 70701459 IC50 > 40000 nM T16042 CGWS12 70701461 IC50 > 25000 nM T16042 CI7Z8X 70701462 IC50 = 460 nM T16042 CQIK83 70701463 IC50 = 3600 nM T16042 C64RVY 70701464 IC50 > 40000 nM T16042 CM34VK 70701465 IC50 = 810 nM T16042 CE04VO 70701466 IC50 > 40000 nM T16042 CQR28O 70701467 IC50 = 5400 nM T16042 CE25CT 70701468 IC50 = 550 nM T16042 CZ0SB3 70701469 IC50 > 30000 nM T16042 C6HB3J 70701472 IC50 > 40000 nM T16042 CH06SB 70701473 IC50 = 23000 nM T16042 C0JU4M 70701475 IC50 > 30000 nM T16042 CZU4X3 70701476 IC50 = 120 nM T16042 CYN9G5 70789634 IC50 > 30000 nM T16042 CF0ZV4 71295953 IC50 > 40000 nM T16042 CTZ59M 71307312 IC50 = 840 nM T16042 CQ28FD 71562304 IC50 >= 50000 nM T16042 CN5RB7 71864212 IC50 = 130 nM T16042 C2OZ9H 72375189 IC50 > 10000 nM T16042 CIK5A0 76321348 IC50 = 5100 nM T16042 CO7KA5 76321349 IC50 = 4500 nM T16042 CN6AE5 76332191 IC50 > 100000 nM T16042 CIS0R8 76335724 IC50 > 10000 nM T16042 CL3XS0 81689867 IC50 > 10000 nM T16042 C79NRZ 86619648 IC50 = 672 nM T16042 C1NM3Q 86619651 IC50 = 855 nM T16042 C12JEM 90643733 IC50 = 8200 nM T16042 CR7UA8 90655993 IC50 = 7600 nM T16042 CR0AW7 122183860 IC50 = 47 nM T16042 CQ2ZR7 122183861 IC50 = 17 nM T16042 CEA49L 122183862 IC50 = 1944 nM T16042 C3Q8VM 122183866 IC50 = 222 nM T16042 CB9T1Z 122185517 IC50 = 39 nM T16042 C1DEB4 122185518 IC50 = 10 nM T16042 CU50CV 122185520 IC50 = 27 nM T16042 C9SK0U 122185521 IC50 = 216 nM T16042 C2U4RI 122192006 Ki = 930 nM T16042 CRTE63 122192007 Ki = 720 nM T16042 C5RZJ7 122192008 Ki = 290 nM T16042 CF8VS9 122192009 Ki = 30 nM T16042 CRB2W6 122192010 Ki = 120 nM T16042 CY7H2X 122192011 Ki = 170 nM T16042 CLTW58 122192012 Ki = 80 nM T16042 CU0CW7 122192013 Ki = 100 nM T16042 C4FYB9 122192014 Ki = 210 nM T16042 CPW97F 122192015 Ki = 830 nM T16042 CNM98J 122192016 Ki = 480 nM T16042 CL34BX 122192017 Ki = 310 nM T16042 CGP4D5 122192018 Ki = 220 nM T16042 CDI32Q 122192019 Ki = 1 nM T16042 CREB46 134132679 IC50 >= 50000 nM T16042 CIB4Q1 134135077 IC50 >= 50000 nM T16042 CI6Z9A 134135690 IC50 > 50000 nM T16042 C2L0QC 134138831 IC50 >= 50000 nM T16042 C1D4GE 134141576 IC50 >= 50000 nM T16042 C2C6WD 134141953 IC50 = 28200 nM T16042 CJC1M8 134142298 IC50 >= 50000 nM T16042 C2EVN5 134142779 IC50 = 47300 nM T16042 CF2GS3 134143695 IC50 = 41500 nM T16042 C02LGE 134144589 IC50 = 25900 nM T16042 CAGV94 134146525 IC50 >= 50000 nM T16042 C8G0DT 134146546 IC50 >= 50000 nM T16042 CJG16L 134148200 IC50 = 15200 nM T16042 C87WBF 134149438 IC50 = 19800 nM T16042 CHKB47 134149557 IC50 > 50000 nM T16042 C4AVJ8 134150456 IC50 = 19000 nM T16042 CNLF02 134152941 IC50 >= 50000 nM T16042 CJQN37 134154892 IC50 > 50000 nM T16042 CDJ50M 134155878 IC50 >= 50000 nM T16042 CE50JR 134158001 IC50 = 17900 nM T16042 CTN03P 136203737 Ki = 23 nM T16042 CSK95Y 136504263 IC50 = 13 nM T16042 C0NE1U 145874872 IC50 = 190 nM T16042 CWJ85C 145949893 IC50 > 100000 nM T16042 C63QRU 145950051 IC50 = 6900 nM T16042 CD08FT 145950994 IC50 = 41800 nM T16042 CSE72B 145951224 IC50 > 100000 nM T16042 C8UYC2 145952049 IC50 = 44100 nM T16042 CL5X8Y 145952410 IC50 = 6300 nM T16042 CN6OZ0 145953984 IC50 > 100000 nM T16042 CI1PG5 145953985 IC50 = 35700 nM T16042 C1YZR4 145954154 IC50 = 39000 nM T16042 CFD28B 145954392 IC50 > 100000 nM T16042 CAZE25 145956011 IC50 = 67900 nM T16042 C0G8YH 145956045 IC50 > 100000 nM T16042 CG0BX5 145956508 IC50 > 100000 nM T16042 C7Z0NR 145957911 IC50 > 100000 nM T16042 CC2K1I 145958434 IC50 = 36100 nM T16042 CUX51R 145958477 IC50 > 100000 nM T16042 C0FJR4 145958570 IC50 = 58200 nM T16042 C8ZW0V 145958955 IC50 = 8300 nM T16042 CL2U5O 145959396 IC50 = 13200 nM T16042 COD91Z 145971498 IC50 > 100000 nM T16042 CE9W5C 145973831 IC50 = 11800 nM T16042 C0V1ON 145978646 IC50 > 100000 nM T16042 CPB8R9 154706252 IC50 = 230 nM T16042 CZTR26 155510499 IC50 > 10000 nM T16042 C1W8QO 155513769 IC50 = 5810 nM T16042 CK41HW 155513870 IC50 > 10000 nM T16042 CIEO91 155515291 IC50 = 740 nM T16042 CF72NM 155515589 IC50 = 2870 nM T16042 C27ZTX 155516046 IC50 = 2950 nM T16042 CB6YH2 155516476 IC50 > 20000 nM T16042 C1LN6S 155516653 IC50 = 2430 nM T16042 CT1N8J 155517121 IC50 > 10000 nM T16042 CJIX40 155519827 IC50 > 10000 nM T16042 CZ7P5Q 155523189 IC50 > 20000 nM T16042 CR8M2G 155526566 IC50 > 20000 nM T16042 CM6BW4 155528084 IC50 > 10000 nM T16042 C0RN3F 155529245 IC50 = 4220 nM T16042 CKO7H8 155533087 IC50 = 740 nM T16042 CLT7B4 155533515 IC50 = 990 nM T16042 CFI01H 155533565 IC50 > 10000 nM T16042 CJA8Q1 155534099 IC50 > 20000 nM T16042 CEOY34 155536295 IC50 = 470 nM T16042 CXV14L 155536874 IC50 = 780 nM T16042 C2P5TI 155539323 IC50 = 750 nM T16042 CVD8P2 155542466 IC50 = 140 nM T16042 C83NFL 155547600 IC50 > 10000 nM T16042 C20GSU 155551132 IC50 > 10000 nM T16042 CF6RY7 155552537 IC50 = 920 nM T16042 CH9M4T 155554130 IC50 = 400 nM T16042 CARW30 155554227 IC50 > 20000 nM T16042 CY16PH 155554639 IC50 = 1290 nM T16042 CJ8BZ2 155554651 IC50 = 1800 nM T16042 C3P6RJ 155557748 IC50 > 10000 nM T16042 C8H4DQ 155560752 IC50 > 10000 nM T16042 CNO28B 155562426 IC50 > 20000 nM T16042 C08OSE 155562991 IC50 > 10000 nM T16042 CY5C0M 155563974 IC50 = 270 nM T16042 CC65QI 155565216 IC50 = 190 nM T16042 CU2C8H 155568009 IC50 > 10000 nM T16042 D00YEV 5281605 Ki = 600 nM T16042 D01KKU 5281894 IC50 > 100000 nM T16042 D03NLE 9947690 IC50 = 17000 nM T16042 D03YMX 11093078 IC50 = 5000 nM T16042 D04JWS 324974 IC50 > 25000 nM T16042 D05FJM 460087 IC50 = 7000 nM T16042 D05HOO 7244 IC50 > 100000 nM T16042 D06PRC 5281650 IC50 = 3100 nM T16042 D06YGF 5281787 IC50 = 130 nM T16042 D07EAJ 10110469 IC50 = 300 nM T16042 D07EGB 3610 IC50 > 10000 nM T16042 D07JRW 10179787 IC50 = 1400 nM T16042 D07ODE 680935 IC50 = 47 nM T16042 D08WDW 10007601 Ki = 8000 nM T16042 D0A5BH 10874329 IC50 = 500 nM T16042 D0A8OW 44584380 IC50 = 14500 nM T16042 D0B5GC 11349 IC50 = 73000 nM T16042 D0C3AG 11978695 IC50 = 7400 nM T16042 D0F1VR 44396194 IC50 = 11000 nM T16042 D0F9FG 46907602 IC50 = 5300 nM T16042 D0H8FG 637821 IC50 = 1700 nM T16042 D0I6ZS 476857 IC50 = 580 nM T16042 D0JL2T 5393152 IC50 > 100000 nM T16042 D0K0QU 11740143 IC50 = 7200 nM T16042 D0L6RV 3086109 IC50 = 15000 nM T16042 D0M6KL 11211821 IC50 = 48000 nM T16042 D0M9VY 23662099 IC50 = 900 nM T16042 D0MF5Y 5281614 IC50 = 1400 nM T16042 D0NQ7I 10029508 IC50 = 900 nM T16042 D0NU1W 636835 IC50 = 800 nM T16042 D0P1LP 7090 IC50 = 420 nM T16042 D0Q0LD 15482063 Ki > 500000 nM T16042 D0US4S 5283159 IC50 > 25000 nM T16042 D0V1DW 11952901 IC50 = 7400 nM T16042 D0X4BT 425241 IC50 = 9400 nM T16042 D0X4CI 9986835 IC50 = 700 nM T11241 D07UHS 107970 EC50 = 3 nM T11241 D07FKQ 44599207 EC50 = 5000 nM T11241 D07UGA 5283560 IC50 = 0.04 nM T11241 D0I2RB 11502996 Ki > 5630 nM T11241 D0L9KH 44623998 EC50 > 10000 nM T11241 D0Y4SI 11363176 EC50 = 109 nM T11241 D04NEO 25031140 EC50 = 46 nM T11241 D04UXN 25182901 EC50 = 3270 nM T11241 D0EP8Y 86299710 EC50 = 2600 nM T11241 D0HW8T 76325532 EC50 = 757 nM T11241 D0K4BI 10223146 IC50 > 1000 nM T11241 D0PW0R 71547555 IC50 > 10000 nM T11241 D0R7ED 76325522 EC50 = 736 nM T11241 C3RZ6P 904918 EC50 > 10000 nM T11241 C1E4SA 1009742 EC50 > 25000 nM T11241 CNEX97 2727676 IC50 = 15670 nM T11241 CCJ2E1 2727678 IC50 = 11600 nM T11241 CPO6B9 2740144 IC50 > 10000 nM T11241 CN29JD 2799937 IC50 > 5000 nM T11241 CE2LQ9 3212803 EC50 > 10000 nM T11241 CZ9UI1 3212804 EC50 > 10000 nM T11241 C4WI2Z 3212805 EC50 > 10000 nM T11241 CS1PB7 3212808 EC50 > 10000 nM T11241 C2HP3Z 3212809 EC50 > 10000 nM T11241 C2ZH6U 3245758 EC50 = 6595 nM T11241 CRZ85P 3721977 EC50 > 10000 nM T11241 C7N5UR 4107292 IC50 > 10000 nM T11241 CAS36H 4460714 IC50 = 8750 nM T11241 CIA43B 4492589 IC50 > 20000 nM T11241 CV69WH 5307570 EC50 > 50000 nM T11241 C89ATE 5309153 EC50 = 434 nM T11241 CZE96X 6056442 IC50 = 3440 nM T11241 C72DNW 9796603 IC50 = 40 nM T11241 CS8MB9 9821227 EC50 = 50.8 nM T11241 C1K9GW 9824415 IC50 = 8200 nM T11241 CHB81X 9883039 IC50 = 9700 nM T11241 CW37CN 9969355 EC50 = 4200 nM T11241 C7FGR9 9979368 IC50 = 12000 nM T11241 CI3K9Z 10023913 EC50 = 89 nM T11241 CZLT30 10045980 IC50 > 10000 nM T11241 C9EK7H 10086559 IC50 = 13050 nM T11241 CA4HX3 10125861 IC50 = 14 nM T11241 C8KXE2 10125862 IC50 = 370 nM T11241 CG6O1W 10125882 IC50 = 350 nM T11241 C7B8UT 10126584 IC50 = 4.9 nM T11241 CG65LQ 10126736 IC50 = 74 nM T11241 CN8H2S 10127475 IC50 = 530 nM T11241 CCG97S 10127776 IC50 = 2100 nM T11241 CGCK28 10149985 IC50 = 2.7 nM T11241 CO06YT 10150171 IC50 = 0.71 nM T11241 C3LG4R 10150372 IC50 = 6 nM T11241 CPU38H 10151146 IC50 = 13 nM T11241 CE9WX6 10172338 IC50 = 280 nM T11241 CDE1S4 10172354 IC50 = 8.5 nM T11241 CI5X6K 10172513 IC50 = 260 nM T11241 CWJO04 10172546 IC50 = 1.1 nM T11241 CS62VA 10173002 IC50 = 1000 nM T11241 CL2QV0 10173327 IC50 = 610 nM T11241 CSV6Q3 10174181 IC50 = 830 nM T11241 C5XFN7 10174255 EC50 = 17 nM T11241 C8XZV1 10174548 IC50 = 430 nM T11241 CG3DX8 10193676 IC50 = 390 nM T11241 CR9YM8 10193915 IC50 = 1.2 nM T11241 C5HJB9 10195325 IC50 = 1000 nM T11241 CY1T7W 10215138 IC50 = 10 nM T11241 C56XBS 10215741 IC50 = 280 nM T11241 CN2FJ9 10216035 IC50 = 130 nM T11241 C6NP8S 10217498 IC50 = 2000 nM T11241 C9KH2F 10236683 IC50 = 1200 nM T11241 CN93ZD 10249887 IC50 = 12000 nM T11241 C6H9VI 10249979 IC50 > 10000 nM T11241 C2O4UR 10251062 IC50 > 10000 nM T11241 C2YZC3 10271422 IC50 = 510 nM T11241 CN0EC2 10286857 IC50 = 170 nM T11241 CKPV49 10287091 IC50 = 110 nM T11241 C74CKG 10287343 IC50 = 99 nM T11241 CW5JG7 10287365 IC50 = 180 nM T11241 C3R1AI 10288370 IC50 > 10000 nM T11241 C5MDF6 10288527 IC50 = 7500 nM T11241 C6EY2U 10289318 IC50 = 94 nM T11241 CJ26CW 10308738 IC50 = 170 nM T11241 C2U3LT 10309022 IC50 = 7600 nM T11241 C8VP3G 10309271 IC50 = 110 nM T11241 C7B2FU 10309462 IC50 = 44 nM T11241 CAF85E 10310253 IC50 = 26 nM T11241 CPK61C 10310952 IC50 > 10000 nM T11241 C8HBY4 10311227 IC50 = 200 nM T11241 C3SM5Z 10317453 IC50 = 58000 nM T11241 CG89DO 10363915 IC50 = 3.86 nM T11241 CDV3W7 10384596 IC50 = 18 nM T11241 C8WL6R 10408874 IC50 = 14000 nM T11241 COQ65E 10409838 IC50 > 10000 nM T11241 CI3EW1 10430549 IC50 = 12 nM T11241 CAL72D 10476387 IC50 ~ 10000 nM T11241 C9NRD6 11168252 IC50 > 10000 nM T11241 CD8T1W 11222939 EC50 = 1.7 nM T11241 CUR1P8 11224984 EC50 = 105 nM T11241 CFPH94 11248292 IC50 = 2100 nM T11241 CK65MP 11271470 IC50 = 4300 nM T11241 C6N4UQ 11280849 EC50 > 10000 nM T11241 CVJX85 11313781 EC50 = 3300 nM T11241 C9JZP8 11315069 EC50 = 114 nM T11241 C34OBY 11315717 EC50 > 10000 nM T11241 C6ZFY8 11315809 EC50 = 3200 nM T11241 COS3Y2 11360553 EC50 = 1200 nM T11241 CAS3N4 11371585 EC50 = 3300 nM T11241 C6JX5O 11397995 EC50 = 7200 nM T11241 C69NSZ 11405953 EC50 = 6700 nM T11241 C9NOJ7 11406331 EC50 > 10000 nM T11241 CYH0U8 11408903 IC50 = 10000 nM T11241 CER35T 11466640 IC50 > 10000 nM T11241 C1SMT3 11484624 EC50 = 9000 nM T11241 CP45BX 11495124 EC50 = 5200 nM T11241 CW51YT 11495139 IC50 > 1000 nM T11241 CDE78J 11496072 EC50 = 184 nM T11241 CWL71C 11496105 EC50 = 9300 nM T11241 CS5A1E 11501417 IC50 = 10000 nM T11241 C7EOU1 11501764 IC50 > 1000 nM T11241 CR1ME9 11501873 EC50 = 4070 nM T11241 CS27OX 11502026 IC50 > 10000 nM T11241 CDVR16 11503306 EC50 = 4000 nM T11241 CL50IH 11503967 EC50 > 3000 nM T11241 CC02BK 11510741 IC50 = 100 nM T11241 CS4LD8 11530826 EC50 > 10000 nM T11241 CK0Y6I 11531691 EC50 > 10000 nM T11241 CQ6S5W 11531879 EC50 > 30000 nM T11241 CAG0Y9 11540052 EC50 = 47.3 nM T11241 CTF1L4 11553135 EC50 > 10000 nM T11241 CU0C3H 11553524 EC50 = 1350 nM T11241 CR5ED7 11555202 IC50 = 160 nM T11241 CLP3O7 11567535 EC50 = 2780 nM T11241 C52ZWY 11568129 EC50 = 623 nM T11241 C3BK8V 11568622 EC50 > 30000 nM T11241 CVW6Q3 11575787 IC50 = 4018 nM T11241 CB75ZP 11575913 EC50 = 230 nM T11241 C5NAQ2 11589375 EC50 = 879 nM T11241 C02XSU 11595314 EC50 > 10000 nM T11241 C9F4YI 11597340 EC50 = 4250 nM T11241 CXS54Q 11603220 IC50 > 10000 nM T11241 C5BDY3 11603528 EC50 > 10000 nM T11241 CCW90K 11603726 EC50 = 940 nM T11241 C96LNP 11604577 IC50 = 4282 nM T11241 CAN4Q9 11611053 EC50 = 470 nM T11241 C7I6ZU 11619303 EC50 > 30000 nM T11241 C41XAE 11624780 EC50 = 1200 nM T11241 CCY7J2 11626664 EC50 = 160 nM T11241 C4IMA6 11632823 EC50 > 10000 nM T11241 CXZ8T6 11633613 EC50 = 2200 nM T11241 CA8W5N 11646599 EC50 = 460 nM T11241 C21VTL 11647892 EC50 > 1000 nM T11241 CYS5F1 11653967 IC50 > 10000 nM T11241 C8TL6P 11654374 EC50 > 10000 nM T11241 CMJ32O 11662328 EC50 = 400 nM T11241 CQTW52 11675496 EC50 > 10000 nM T11241 C8CQ2N 11675907 EC50 = 780 nM T11241 CD4AO7 11676168 EC50 = 350 nM T11241 CCNU48 11678855 EC50 = 31.62 nM T11241 CR94XU 11682224 EC50 > 10000 nM T11241 C3Q9JR 11682677 EC50 = 330 nM T11241 CVG41H 11682696 EC50 = 620 nM T11241 CQRA36 11683935 IC50 = 21.1 nM T11241 CCF80W 11689680 EC50 = 110 nM T11241 CTB2W7 11690483 EC50 = 489 nM T11241 C8XLO4 11690779 IC50 = 628 nM T11241 C0BR1U 11696807 IC50 > 10 nM T11241 CK5S1L 11697013 EC50 = 950 nM T11241 CL80RC 11697277 EC50 = 1800 nM T11241 C2ZWP0 11697911 EC50 = 51 nM T11241 CK63OB 11705484 IC50 = 10000 nM T11241 C4G2OP 11743459 IC50 = 13000 nM T11241 CZ6YN9 11752659 IC50 > 10000 nM T11241 CJ98PB 11852048 EC50 > 10000 nM T11241 CV3WI7 11852049 EC50 = 4447 nM T11241 C2Z8AY 11852142 EC50 = 4450 nM T11241 C3J8TH 11852143 EC50 = 1400 nM T11241 C2FEG4 11852144 EC50 = 1098 nM T11241 CRVF18 11852146 EC50 > 10000 nM T11241 CLI76U 11852148 EC50 > 10000 nM T11241 CEW5F3 11852233 EC50 = 569 nM T11241 C9D3UE 11852234 EC50 = 1755 nM T11241 C0J2EH 11852237 EC50 = 40.6 nM T11241 C67GNU 11852437 EC50 = 126 nM T11241 CWF0P2 11852636 EC50 = 8558 nM T11241 CI1S6O 11852848 EC50 = 314 nM T11241 CB67GQ 11852952 EC50 = 392 nM T11241 CH5W6S 11852953 EC50 = 4418 nM T11241 CUBD18 11852955 EC50 = 122 nM T11241 C4N3DG 11853337 EC50 = 780 nM T11241 CMK7W8 11853338 EC50 = 2840 nM T11241 CQ0V5W 11853576 EC50 = 1040 nM T11241 C7YJM4 11853579 EC50 = 8420 nM T11241 C09ZXI 11853580 EC50 = 201 nM T11241 CFUQ37 11853832 EC50 = 7470 nM T11241 CU6M7E 11853834 EC50 = 597 nM T11241 CWR71V 11853835 EC50 = 1000 nM T11241 CMJ71A 11853836 EC50 = 875 nM T11241 CKOR74 11854090 EC50 = 3410 nM T11241 CQ78BJ 11854356 EC50 = 566 nM T11241 CS8E1K 11854607 EC50 = 430 nM T11241 CF7W9B 11854857 EC50 = 555 nM T11241 CLHA36 11869937 EC50 > 1000 nM T11241 C1LMA8 11977818 EC50 = 900 nM T11241 CA9D8B 11977936 EC50 > 20000 nM T11241 C03OUS 11977938 EC50 > 20000 nM T11241 CUM5T9 11977939 EC50 > 20000 nM T11241 CYE48W 11978048 EC50 = 15000 nM T11241 CPSI96 11978050 EC50 > 20000 nM T11241 CGS70F 11978162 EC50 > 20000 nM T11241 COY96U 11978278 EC50 > 20000 nM T11241 CDI32A 16038017 EC50 = 1600 nM T11241 CE5OB2 16051482 EC50 > 5000 nM T11241 C4TQR8 16105530 IC50 = 2960 nM T11241 CW1QC9 16105531 IC50 = 11390 nM T11241 C4MZ2T 16105532 IC50 = 13230 nM T11241 C8IBY5 16105533 IC50 = 9740 nM T11241 CJ2E4B 16105541 IC50 = 3570 nM T11241 C65RDB 16188020 EC50 > 50000 nM T11241 CLA85D 16657820 EC50 = 74 nM T11241 CX71MV 16735046 EC50 > 25000 nM T11241 CS0X4J 16736754 EC50 = 4800 nM T11241 CG8J5U 16736755 EC50 = 10300 nM T11241 CA9P2L 16737316 EC50 > 25000 nM T11241 C6FW1V 16737319 EC50 > 25000 nM T11241 CC6W8M 16737345 EC50 = 1440 nM T11241 CY7U2O 16737504 EC50 = 1900 nM T11241 CR0B6Y 16737505 EC50 > 25000 nM T11241 C58EWF 16737507 EC50 = 3430 nM T11241 CU30WQ 16737509 EC50 > 25000 nM T11241 CZ41LC 16737511 EC50 > 25000 nM T11241 C4D2EF 16737513 EC50 = 25000 nM T11241 CU6Y0F 16737514 EC50 > 25000 nM T11241 CF4XN8 16737667 EC50 > 25000 nM T11241 C6X5BR 16737668 EC50 > 4300 nM T11241 C6M2FB 16737670 EC50 > 25000 nM T11241 CDG57C 16737679 EC50 = 1730 nM T11241 CIJF78 16737988 EC50 > 10000 nM T11241 CRE74S 16738333 EC50 > 25000 nM T11241 CGAD08 17253208 EC50 = 105 nM T11241 CIEK03 17253281 EC50 = 959 nM T11241 C6HB9A 21455530 IC50 = 15 nM T11241 CNV98Q 23121057 EC50 > 10000 nM T11241 C89BVX 23121067 EC50 > 10000 nM T11241 CC75ZH 23121172 EC50 = 3000 nM T11241 C0O5CY 23121189 EC50 = 5500 nM T11241 CLZ45N 23121209 EC50 > 10000 nM T11241 C6DV2O 23121326 EC50 > 30000 nM T11241 C7XK3S 23121338 EC50 = 7800 nM T11241 CK6G0D 23121374 EC50 = 1900 nM T11241 CI7RA6 23121393 EC50 > 30000 nM T11241 C05RUE 23121412 EC50 > 10000 nM T11241 C6MJ4N 23121431 EC50 > 10000 nM T11241 CF01WY 23121435 EC50 = 7200 nM T11241 CME14G 23121436 EC50 > 10000 nM T11241 C5AKM6 23121505 EC50 > 30000 nM T11241 C14XBN 23121526 EC50 > 10000 nM T11241 CF1EU4 23121592 EC50 > 10000 nM T11241 CYX03D 23121622 EC50 > 10000 nM T11241 CUF57G 23729211 EC50 = 236 nM T11241 CEV1I3 23729229 EC50 = 528 nM T11241 C8R4SV 24744028 EC50 > 3000 nM T11241 C2JGS9 24784418 EC50 = 320 nM T11241 C6I0ED 24812110 IC50 = 6.3 nM T11241 C0O9UG 24825338 EC50 = 110 nM T11241 CB82GW 24825339 EC50 = 2760 nM T11241 CTH4S8 24850258 EC50 = 1110 nM T11241 C9QTZ3 24851764 EC50 = 1710 nM T11241 CW2CD1 24851766 EC50 = 519 nM T11241 CU79ZI 24956673 EC50 = 120 nM T11241 C3RPZ4 24956674 EC50 = 189 nM T11241 CF9I1S 24956675 EC50 = 139 nM T11241 CYIJ40 24956676 EC50 = 264 nM T11241 CPT9J2 24957028 EC50 = 129 nM T11241 CU3R0D 24957029 EC50 = 81 nM T11241 C90SNU 24986381 EC50 > 10000 nM T11241 C95TGD 24986921 EC50 > 20000 nM T11241 C1TGE9 25008420 IC50 = 2000 nM T11241 CV6EP4 25008421 EC50 > 3000 nM T11241 C34RKU 25031771 EC50 = 1532 nM T11241 CCJ17D 25032056 EC50 = 310 nM T11241 C9WQC5 25072410 EC50 = 307 nM T11241 CCO54A 25074253 EC50 = 350 nM T11241 CLT95X 25110105 EC50 > 50000 nM T11241 CLW5E6 25110210 EC50 = 7000 nM T11241 CUZJ62 25110212 EC50 = 6563 nM T11241 C14EAK 25110484 EC50 = 323 nM T11241 C3S8QZ 25110485 EC50 = 1375 nM T11241 C01FRW 25110488 EC50 = 103 nM T11241 C07GXT 25110489 EC50 = 7985 nM T11241 CAP8T1 25110492 EC50 = 1683 nM T11241 CWUT04 25110494 EC50 = 3430 nM T11241 CXU68J 25110496 EC50 = 202 nM T11241 CI2VH9 25110498 EC50 = 337 nM T11241 CLEF36 25110499 EC50 = 535 nM T11241 C8WAX0 25110500 EC50 = 3536 nM T11241 CS2WQ0 25110501 EC50 = 2820 nM T11241 CF50YO 25110510 EC50 = 1740 nM T11241 CJ3HS1 25110511 EC50 = 2753 nM T11241 CJ9CI6 25110521 EC50 > 50000 nM T11241 CP6A9Q 25110522 EC50 > 50000 nM T11241 C14CBE 25110524 EC50 > 50000 nM T11241 C1EM2P 25154344 EC50 = 62 nM T11241 C6RM3T 25182621 EC50 > 30000 nM T11241 C1HT8Z 25182756 EC50 > 30000 nM T11241 CP1CA9 25182769 EC50 > 30000 nM T11241 CF35EH 25182773 EC50 > 30000 nM T11241 C0Y2ZH 25182781 EC50 > 30000 nM T11241 CGEM35 25182899 EC50 = 416 nM T11241 CNYW93 25182926 EC50 = 1094 nM T11241 C10HKX 25192001 EC50 = 0.215 nM T11241 CL7RV5 25192005 EC50 = 0.15 nM T11241 CB06TP 25192006 EC50 > 5000 nM T11241 CZ8Y9S 42610387 EC50 > 10000 nM T11241 CHD3I5 42622931 EC50 = 120 nM T11241 C48TPJ 42630194 EC50 > 100000 nM T11241 C9YBE0 42636433 EC50 = 10000 nM T11241 CA81LQ 42636536 EC50 = 25118.86 nM T11241 CS35FG 42636618 EC50 > 31622.78 nM T11241 CNHI02 44124898 EC50 = 15848.93 nM T11241 CDL1C8 44125170 EC50 > 31622.78 nM T11241 CG5X4T 44125468 EC50 > 31622.78 nM T11241 CNU5F1 44125469 EC50 = 7943.28 nM T11241 CH3A1V 44125470 EC50 = 1995.26 nM T11241 C51WHA 44125471 EC50 > 31622.78 nM T11241 CRE0O1 44125588 EC50 = 794.33 nM T11241 CP1BF0 44125589 EC50 = 251.19 nM T11241 CS0H1B 44125704 EC50 = 10000 nM T11241 C1YHG6 44128660 EC50 > 31622.78 nM T11241 C4H5TR 44128662 EC50 > 31622.78 nM T11241 CUQE25 44128745 EC50 = 7943.28 nM T11241 CAH09Q 44128746 EC50 > 31622.78 nM T11241 C31VJX 44128747 EC50 > 31622.78 nM T11241 C7H4MR 44128748 EC50 > 31622.78 nM T11241 CH2ES5 44128819 EC50 > 31622.78 nM T11241 CRIK86 44128821 EC50 > 31622.78 nM T11241 CIL7J3 44128904 EC50 > 31622.78 nM T11241 CY83JW 44128905 EC50 > 31622.78 nM T11241 C19YHX 44128909 EC50 = 1995.26 nM T11241 C47OXT 44128987 EC50 = 7943.28 nM T11241 CW1DL9 44129063 EC50 > 31622.78 nM T11241 CN5O1Y 44129065 EC50 > 31622.78 nM T11241 CCTS05 44129140 EC50 = 6309.57 nM T11241 CTV36P 44129142 EC50 = 15848.93 nM T11241 CHL90M 44129143 EC50 > 31622.78 nM T11241 C4EP2M 44129144 EC50 = 1995.26 nM T11241 CP6MQ2 44129145 EC50 = 25118.86 nM T11241 CABP65 44129218 EC50 > 31622.78 nM T11241 C1BT4A 44129293 EC50 > 31622.78 nM T11241 CAQ28H 44129298 EC50 = 5011.87 nM T11241 CY1X3Z 44129373 EC50 = 12589.25 nM T11241 CG73ST 44138103 EC50 > 100000 nM T11241 CVUJ04 44199411 EC50 = 425 nM T11241 CNJ96W 44199424 EC50 = 125 nM T11241 C47CJM 44199450 EC50 = 616 nM T11241 CLR62S 44217168 EC50 = 910 nM T11241 CD3IM6 44217169 EC50 = 570 nM T11241 CC43PQ 44217170 EC50 = 3200 nM T11241 C58BOP 44217502 EC50 = 8 nM T11241 C75XPC 44217654 EC50 = 3.5 nM T11241 CEHB49 44217839 EC50 = 139 nM T11241 CH0VO9 44217997 EC50 = 1400 nM T11241 C7CB5P 44218002 EC50 = 154 nM T11241 C5L0QT 44218130 EC50 = 1.4 nM T11241 CO41AS 44218131 EC50 = 480 nM T11241 CI34VL 44218450 EC50 = 100 nM T11241 CWIC07 44218451 EC50 = 4300 nM T11241 C7B1PL 44218479 EC50 = 520 nM T11241 C4F6RA 44218604 EC50 = 30 nM T11241 C25HOP 44218903 EC50 = 176 nM T11241 CWNE68 44219368 EC50 = 2000 nM T11241 C8AC7D 44219369 EC50 = 1250 nM T11241 CKYJ71 44219370 EC50 = 380 nM T11241 CJ7M3E 44219525 EC50 = 100 nM T11241 CAY2S1 44219528 EC50 = 350 nM T11241 CH8CM7 44341291 IC50 = 320 nM T11241 CQR2G1 44341399 IC50 = 720 nM T11241 C95GIJ 44342175 Ki = 300 nM T11241 C8NOT7 44342221 EC50 = 845.4 nM T11241 CCN68O 44342231 EC50 = 878.6 nM T11241 CXJ08Y 44342244 EC50 = 862.4 nM T11241 C6LT8S 44342246 EC50 = 601.9 nM T11241 CLXY90 44342331 EC50 = 740 nM T11241 CAUQ90 44342468 EC50 = 1500 nM T11241 CMKZ19 44344194 IC50 = 2.8 nM T11241 CLQ25X 44344210 IC50 = 13 nM T11241 C31BXA 44344270 IC50 = 46 nM T11241 CY7FC4 44344298 IC50 = 55 nM T11241 C1SP9M 44344338 IC50 = 1000 nM T11241 C2D5LZ 44344360 IC50 = 1000 nM T11241 CT4NW0 44344390 IC50 = 0.91 nM T11241 C9S2FH 44344404 IC50 = 2.7 nM T11241 CY9C1D 44344412 IC50 = 14 nM T11241 CLDU29 44344413 IC50 = 4.3 nM T11241 C91OKY 44344446 IC50 = 47 nM T11241 CL3CT8 44344456 IC50 = 2 nM T11241 CS5Z1P 44361546 IC50 > 20000 nM T11241 CJ36UD 44394116 IC50 = 9.8 nM T11241 C5KA6D 44394117 IC50 = 1200 nM T11241 CU7L0K 44394153 IC50 = 19 nM T11241 CT8UN6 44394161 IC50 = 410 nM T11241 C9E6CF 44394169 IC50 = 190 nM T11241 C8H0XM 44394191 IC50 = 2.7 nM T11241 CH2A5S 44394211 IC50 = 51 nM T11241 CND39O 44394212 IC50 = 7 nM T11241 C84JPI 44394247 IC50 = 220 nM T11241 CA28OJ 44394273 IC50 = 4.7 nM T11241 CO0T1E 44394279 IC50 = 5.2 nM T11241 CL5BC6 44394330 IC50 = 220 nM T11241 CI75GS 44398012 EC50 = 1600 nM T11241 CCFT02 44398049 EC50 = 790 nM T11241 CRYM50 44398058 EC50 = 1700 nM T11241 C4DIT3 44398076 EC50 = 630 nM T11241 C3H2IY 44398170 EC50 = 690 nM T11241 CL5SY3 44398172 EC50 = 2700 nM T11241 CR4TH0 44406004 EC50 = 0.1778 nM T11241 C3JF1Q 44406009 EC50 = 5.012 nM T11241 CK6J2H 44406749 EC50 = 19.95 nM T11241 CDY46P 44412165 IC50 = 3800 nM T11241 CR2DT4 44412221 IC50 > 10000 nM T11241 CRV34X 44412232 IC50 = 10000 nM T11241 CV63YC 44412233 IC50 > 10000 nM T11241 CQ1V3J 44412282 IC50 > 10000 nM T11241 CB6KR7 44412294 IC50 > 10000 nM T11241 CTV5M0 44412353 IC50 = 7600 nM T11241 CN7K2O 44412364 IC50 = 2200 nM T11241 CL1GJ3 44412415 IC50 = 6700 nM T11241 CV28IK 44412416 IC50 = 1700 nM T11241 CBM50W 44412428 IC50 > 10000 nM T11241 C2US0I 44412578 EC50 > 10000 nM T11241 CM46YR 44412604 EC50 > 10000 nM T11241 C1LTZ6 44412605 EC50 > 10000 nM T11241 C28CAY 44412621 EC50 > 10000 nM T11241 C9I7UV 44412622 EC50 > 10000 nM T11241 CNF3Y2 44412623 EC50 > 10000 nM T11241 CG7T1N 44412643 EC50 > 10000 nM T11241 C05TUB 44412658 EC50 > 10000 nM T11241 CH51GD 44412659 EC50 > 10000 nM T11241 C93OLQ 44412660 EC50 > 10000 nM T11241 C0CA6R 44412661 EC50 > 10000 nM T11241 CL54DN 44412674 EC50 > 10000 nM T11241 C3M5SO 44412702 EC50 > 1000 nM T11241 CBUQ92 44412827 EC50 = 1220 nM T11241 CBL87K 44412867 EC50 = 460 nM T11241 COA6Q1 44412868 EC50 > 10000 nM T11241 C80JSN 44412882 EC50 = 160 nM T11241 C2WV6S 44412883 EC50 = 1100 nM T11241 C84PLZ 44412908 EC50 > 10000 nM T11241 C78DOK 44412936 EC50 = 470 nM T11241 CH6Z8V 44412962 EC50 > 10000 nM T11241 C3MWD4 44412971 EC50 = 500 nM T11241 CJC06H 44412994 EC50 = 340 nM T11241 CT6EU7 44413274 IC50 = 4800 nM T11241 CYO6R3 44413349 IC50 = 690 nM T11241 CH9NL4 44413365 IC50 = 460 nM T11241 CW8E0R 44413415 IC50 = 2100 nM T11241 CYW5D3 44413430 IC50 = 1500 nM T11241 CJ5S2H 44413446 IC50 > 1000 nM T11241 CWRZ40 44413447 IC50 = 3100 nM T11241 CVC61G 44413482 IC50 > 1000 nM T11241 CN42SQ 44419094 IC50 = 4600 nM T11241 CR4KE6 44419095 IC50 = 3590 nM T11241 CEQ5U3 44419099 IC50 > 20000 nM T11241 CWL92R 44422573 EC50 = 270 nM T11241 C4MTP5 44422590 EC50 = 15000 nM T11241 C0I3LB 44422601 EC50 = 43 nM T11241 C2O7AP 44422604 EC50 = 23 nM T11241 C7O0PC 44422606 EC50 = 100 nM T11241 C2WEQ7 44437392 IC50 = 13000 nM T11241 CP1FN6 44437417 IC50 = 5000 nM T11241 C0W3FQ 44439850 EC50 = 123 nM T11241 CB4Z3I 44439851 EC50 = 2600 nM T11241 C9SFT8 44439852 EC50 > 1000 nM T11241 CS9H0L 44517795 EC50 > 100000 nM T11241 CQF0I7 44547175 EC50 > 10000 nM T11241 C0NMA9 44547315 EC50 > 10000 nM T11241 C5WQ8J 44547316 EC50 > 10000 nM T11241 CJNM95 44547318 EC50 > 10000 nM T11241 CX13MK 44547414 EC50 = 3100 nM T11241 CGZ84E 44547461 EC50 > 10000 nM T11241 CG6D3L 44547603 EC50 > 10000 nM T11241 CU3V6A 44547605 EC50 > 10000 nM T11241 CFI6C1 44547606 EC50 > 10000 nM T11241 C5S0MH 44547608 EC50 > 10000 nM T11241 C27WLJ 44547758 EC50 > 10000 nM T11241 CL2RF3 44547909 EC50 > 10000 nM T11241 CXMF34 44547910 EC50 > 10000 nM T11241 C2OM1R 44547911 EC50 > 10000 nM T11241 CH4F0V 44548058 EC50 > 10000 nM T11241 C46GZY 44548059 EC50 > 10000 nM T11241 CF1JW9 44548061 EC50 > 10000 nM T11241 CMYZ28 44548224 EC50 > 10000 nM T11241 CV9GB5 44548226 EC50 > 10000 nM T11241 COU3R0 44565595 IC50 = 3750 nM T11241 CP18DA 44565596 IC50 = 100 nM T11241 CO8AD3 44565597 EC50 = 63.3 nM T11241 C75UYT 44565621 IC50 = 120 nM T11241 CS13TE 44565622 IC50 = 31.3 nM T11241 CU1NS0 44565703 IC50 = 2500 nM T11241 CIY08J 44565712 IC50 = 50 nM T11241 C16WTE 44565713 IC50 = 1040 nM T11241 COH39N 44565714 EC50 = 1.38 nM T11241 CB1GT5 44565715 EC50 = 28.8 nM T11241 CAV3F9 44565716 EC50 = 54.8 nM T11241 C76DFZ 44565717 IC50 = 20 nM T11241 CMG7L1 44565738 IC50 = 20 nM T11241 CH8SJ9 44565739 IC50 = 6 nM T11241 CX9AZ4 44591249 EC50 = 16.3 nM T11241 C3NOY0 44591250 EC50 = 10.1 nM T11241 C3TAY6 44591264 EC50 = 9.8 nM T11241 CGCL62 44591265 IC50 = 5.3 nM T11241 C10TGI 44591266 EC50 = 10.8 nM T11241 C92QVU 44599024 EC50 = 1310 nM T11241 CI3L4J 44599683 EC50 > 25000 nM T11241 C0EI2G 44599686 EC50 > 2500 nM T11241 CR1FP6 44599687 EC50 = 7120 nM T11241 CRMO89 44600329 EC50 > 2500 nM T11241 C1GW4T 44600476 EC50 = 888 nM T11241 C5I8AH 44600484 EC50 > 25000 nM T11241 CS3RZ6 44600643 EC50 = 836 nM T11241 CJR1B7 44600645 EC50 = 4670 nM T11241 CB94AO 44601271 EC50 > 25000 nM T11241 C7MJV8 44625666 EC50 = 5900 nM T11241 CKS69U 44625752 EC50 = 1100 nM T11241 CV5GL3 44625753 EC50 = 2600 nM T11241 CZUT65 45376040 EC50 > 2000 nM T11241 C7JFL9 45376041 EC50 = 80 nM T11241 CDV7R4 45376042 EC50 > 16000 nM T11241 CYOW10 45377016 IC50 > 10000 nM T11241 C7D3LB 45377018 IC50 > 10000 nM T11241 CN0A4O 45377161 IC50 > 10000 nM T11241 CR32YA 45377248 EC50 = 400000 nM T11241 C6T4QB 45377662 EC50 = 300 nM T11241 C85SQO 45377797 EC50 = 700 nM T11241 CWQY86 45377937 EC50 = 1000 nM T11241 C9AZ0K 45377938 EC50 = 427000 nM T11241 C8ELI4 45378010 IC50 > 10000 nM T11241 CH0Z5C 45378095 EC50 > 40000 nM T11241 C5P7LK 45378098 EC50 > 4000 nM T11241 C73DCB 46174905 EC50 > 10000 nM T11241 CPU02J 46190696 IC50 > 10000 nM T11241 CVDK53 46204808 EC50 > 1000 nM T11241 C5MX8L 46204811 EC50 > 1000 nM T11241 C78PDO 46205128 EC50 > 1000 nM T11241 C1GEB0 46205132 EC50 > 1000 nM T11241 C96WMQ 46205452 EC50 > 1000 nM T11241 C1YQM5 46205453 EC50 > 1000 nM T11241 C1RV6W 46205455 EC50 > 1000 nM T11241 CV1G4W 46205774 EC50 = 13 nM T11241 CLI75U 46205775 EC50 = 4.1 nM T11241 CDA30X 46206103 EC50 > 1000 nM T11241 COR39P 46206105 EC50 = 4.9 nM T11241 CHOV03 46206106 EC50 > 1000 nM T11241 CQKV71 46206107 EC50 > 1000 nM T11241 C1THR5 46206435 EC50 > 1000 nM T11241 CSTA18 46224712 EC50 > 10000 nM T11241 C4QB8F 46224713 EC50 > 1000 nM T11241 C4HN6L 46224714 EC50 > 10000 nM T11241 CF75RO 46224715 EC50 = 1350 nM T11241 C6R9SJ 46224716 EC50 > 1000 nM T11241 CB56OX 46224767 EC50 = 345 nM T11241 CHC1D9 46224768 EC50 > 1000 nM T11241 C15WRO 46224769 EC50 = 995 nM T11241 CMW59H 46225233 EC50 > 10000 nM T11241 CV5T1F 46225282 EC50 > 10000 nM T11241 CF74HE 46225283 EC50 > 10000 nM T11241 C6XAU7 46225284 EC50 > 10000 nM T11241 CL4H8B 46225285 EC50 > 10000 nM T11241 CQ6WU0 46236268 EC50 = 59 nM T11241 CUE6F1 46236269 EC50 = 96 nM T11241 C4NDW1 46236270 EC50 = 114 nM T11241 C01WTY 46236271 EC50 = 128 nM T11241 CV8LH3 46236272 EC50 = 302 nM T11241 CY75PB 46236273 EC50 = 310 nM T11241 CN8IP7 46236274 EC50 = 162 nM T11241 CEAU68 46236398 EC50 = 118 nM T11241 CI5C6D 46236399 EC50 = 18 nM T11241 CDP2R8 46236400 EC50 = 125 nM T11241 C7OUC4 46236401 EC50 > 10000 nM T11241 CW3H8J 46236402 EC50 = 821 nM T11241 C7I3DZ 46236403 EC50 = 200 nM T11241 COV15E 46236404 EC50 = 88 nM T11241 C5XR6Q 46236517 EC50 = 307 nM T11241 CUN5S8 46236518 EC50 = 350 nM T11241 CZAQ79 46236519 EC50 = 458 nM T11241 CB2PV6 46236520 EC50 = 335 nM T11241 CO2YA0 46236521 EC50 = 425 nM T11241 C9SNG5 46236522 EC50 = 246 nM T11241 CZU24S 46236523 EC50 = 144 nM T11241 CKZ0M4 46236660 EC50 = 428 nM T11241 CJOW38 46236661 EC50 = 514 nM T11241 C3O7UR 46236662 EC50 = 127 nM T11241 C8MO1E 46236663 EC50 = 525 nM T11241 C9YXI2 46236664 EC50 = 228 nM T11241 CQ6K2M 46236665 EC50 = 674 nM T11241 CI69FH 46236666 EC50 = 183 nM T11241 CN2O7F 46236805 EC50 = 212 nM T11241 CG8BV2 46236806 EC50 = 317 nM T11241 C8IF1Z 46236807 EC50 = 95 nM T11241 C46YWF 46236808 EC50 = 99 nM T11241 CWE42H 46236809 EC50 = 50 nM T11241 C8GOC2 46236810 EC50 = 335 nM T11241 CU2F3J 46236811 EC50 = 106 nM T11241 CP0J7W 46236929 EC50 = 1385 nM T11241 CDLX95 46236930 EC50 = 165 nM T11241 C43CIM 46236931 EC50 = 136 nM T11241 CG4O8A 46236932 EC50 = 35 nM T11241 CST73W 46236933 EC50 = 103 nM T11241 CP52YF 46236934 EC50 = 212 nM T11241 C1L6YP 46236935 EC50 > 10000 nM T11241 C1SC0X 46237046 EC50 = 5791 nM T11241 CA7W1B 46237047 EC50 = 2583 nM T11241 CJGE86 46237048 EC50 = 6689 nM T11241 CM3B0H 46237049 EC50 = 86 nM T11241 C23JZF 46237050 EC50 = 59 nM T11241 CV4HT8 46237051 EC50 = 54 nM T11241 CL4R3O 46237052 EC50 = 68 nM T11241 C2RJF5 46237175 EC50 = 240 nM T11241 CSW4X8 46237176 EC50 = 1430 nM T11241 CZKV91 46237177 EC50 = 531 nM T11241 C21EUB 46237178 EC50 = 114 nM T11241 CPT48C 46237179 EC50 = 124 nM T11241 CZ01WY 46237180 EC50 = 174 nM T11241 C3PVA2 46237828 EC50 = 1000 nM T11241 C0J8CN 46238363 EC50 = 140 nM T11241 C8N6IR 46238364 EC50 > 10000 nM T11241 C7Q8XW 46238365 EC50 = 8810 nM T11241 C0Q7IH 46238366 EC50 = 1229 nM T11241 C2M9XO 46835914 EC50 = 2900 nM T11241 C9CR0E 46835922 EC50 = 1600 nM T11241 C2XO4K 46846820 EC50 = 4100 nM T11241 CFH04W 46846899 EC50 = 680 nM T11241 CIO26E 46846900 EC50 = 730 nM T11241 CF41CL 46846901 EC50 = 12000 nM T11241 C6DKO5 46846902 EC50 = 2600 nM T11241 C80DQI 46846904 EC50 = 1900 nM T11241 CEF91N 46846906 EC50 = 1000 nM T11241 CA2W3P 46846912 EC50 = 130 nM T11241 CQ1N4Z 46846913 EC50 = 850 nM T11241 CG3RT7 46846915 EC50 = 6200 nM T11241 CSU08A 46846921 EC50 = 1800 nM T11241 CH8TL1 46847145 EC50 = 2100 nM T11241 CI63SP 46847146 EC50 = 8200 nM T11241 CC5JQ3 46847147 EC50 = 1900 nM T11241 CTKC40 46847148 EC50 = 630 nM T11241 CQY5P8 46866185 EC50 = 300 nM T11241 C6LJ7A 46866186 EC50 > 22000 nM T11241 CLS29B 46872626 IC50 > 10000 nM T11241 CAD23F 46880801 EC50 = 2320 nM T11241 CQZ59G 46881623 EC50 = 236 nM T11241 CW6RX2 46881847 EC50 = 5.4 nM T11241 CAHC81 46881875 EC50 = 151 nM T11241 C0BOR7 46881876 EC50 = 3100 nM T11241 CCS12Z 46881877 EC50 = 6400 nM T11241 C3QMS1 46881912 EC50 = 2400 nM T11241 CY3S0L 46883880 EC50 = 922.1 nM T11241 CTL89X 46884020 EC50 = 0.286 nM T11241 CYJL86 46885693 IC50 > 10000 nM T11241 C17RPW 46885694 IC50 > 10000 nM T11241 C7SB8P 46885695 IC50 > 1000 nM T11241 C1I9TX 46885696 IC50 > 1000 nM T11241 CC60OX 46885742 IC50 = 2000 nM T11241 CEQ7V1 46885743 IC50 = 285 nM T11241 CF5V3E 46885744 IC50 = 1000 nM T11241 COL9E8 46885745 IC50 = 3250 nM T11241 CJ21TY 46885796 EC50 > 3000 nM T11241 CGTR17 46885797 IC50 = 700 nM T11241 CZDL71 46885798 EC50 > 3000 nM T11241 CL0C6G 46885873 EC50 > 1000 nM T11241 CWV3O6 46886019 EC50 = 83 nM T11241 CV6WT1 46929213 EC50 > 10000 nM T11241 C5Z6RM 49839234 EC50 = 10000 nM T11241 CL64TH 49842175 EC50 = 25118.86 nM T11241 CPJ25K 49847296 EC50 > 31622.78 nM T11241 C8KQB9 49848139 EC50 > 10000 nM T11241 CNA18Z 49848426 EC50 > 31622.78 nM T11241 CU86ZT 49848427 EC50 > 31622.78 nM T11241 CAL07G 49848428 EC50 > 31622.78 nM T11241 CJGR71 49848429 EC50 > 31622.78 nM T11241 C29KYX 49848430 EC50 > 31622.78 nM T11241 C4BXP1 49848557 EC50 > 31622.78 nM T11241 CZG98A 49848559 EC50 > 31622.78 nM T11241 CKD3E5 49848560 EC50 > 31622.78 nM T11241 CK29IW 49848561 EC50 > 31622.78 nM T11241 CHLR06 49848655 EC50 > 10000 nM T11241 CQ32CR 49848656 EC50 > 10000 nM T11241 C07NGT 49848778 EC50 > 10000 nM T11241 C74KWB 49848898 EC50 > 10000 nM T11241 CMV6Y2 49868651 EC50 = 5300 nM T11241 CA7M0E 49871977 EC50 = 96 nM T11241 CE7I5G 49872065 EC50 = 71 nM T11241 C6QH3P 49872066 EC50 = 690 nM T11241 C7LQ8B 50923120 EC50 = 12000 nM T11241 CT56SE 50923123 EC50 = 4500 nM T11241 CDG10V 50923126 EC50 = 1800 nM T11241 CH10BV 50923273 EC50 = 1300 nM T11241 CFQV13 50923275 EC50 = 2000 nM T11241 C69IWK 50923276 EC50 = 21000 nM T11241 CD75CR 50923423 EC50 = 20300 nM T11241 CU62PH 50923424 EC50 = 900 nM T11241 C8X0ZH 50923425 EC50 = 5600 nM T11241 CC2VU3 50923427 EC50 = 12000 nM T11241 CBL82V 50925335 EC50 > 31300 nM T11241 CNM61U 50925336 EC50 = 1200 nM T11241 CH0B8K 50925337 EC50 = 9400 nM T11241 CVDN46 51346809 EC50 > 10000 nM T11241 C2W8LE 51346934 EC50 = 3470 nM T11241 C48OFS 53317713 EC50 = 542 nM T11241 CFL29U 53318124 EC50 = 1210 nM T11241 C6QY0V 53318125 EC50 = 2890 nM T11241 CG1KZ7 53318790 EC50 = 6090 nM T11241 CI1D3M 53319457 EC50 = 10100 nM T11241 C45YTZ 53319458 EC50 = 877 nM T11241 CER0W1 53320088 EC50 = 679 nM T11241 CU2P1O 53320107 EC50 = 3880 nM T11241 C9SVK4 53320108 EC50 > 25000 nM T11241 C17BHO 53320170 EC50 > 10000 nM T11241 CWU0X3 53320363 EC50 = 4880 nM T11241 CF3VN5 53322061 EC50 = 478 nM T11241 C5H4NQ 53322110 EC50 > 7200 nM T11241 C56HPB 53322715 EC50 = 354 nM T11241 CA1W8U 53322735 EC50 = 687 nM T11241 CJQ3A1 53322736 EC50 > 25000 nM T11241 CI06MU 53322737 EC50 = 2440 nM T11241 CL14WS 53322738 EC50 = 1800 nM T11241 CG17KO 53323419 EC50 > 25000 nM T11241 C1FXC6 53323420 EC50 = 996 nM T11241 CL4OZ7 53323421 EC50 = 2510 nM T11241 CEP7Z4 53324301 EC50 = 2710 nM T11241 C5TCI2 53324339 EC50 = 1200 nM T11241 CA87QM 53324746 EC50 = 3470 nM T11241 CLHX41 53325368 EC50 > 25000 nM T11241 C7X8YO 53325380 EC50 > 2500 nM T11241 CRA75F 53326036 EC50 > 25000 nM T11241 C7MR1A 53326037 EC50 = 5460 nM T11241 C9T4QX 53326615 EC50 > 25000 nM T11241 CVD5A8 53326641 EC50 = 1910 nM T11241 CQDP84 53326886 EC50 = 967 nM T11241 CC7DZ4 53362086 EC50 > 10000 nM T11241 C9CT8N 53373573 EC50 > 10000 nM T11241 CG3FA9 53492750 EC50 > 31622.78 nM T11241 CW69RX 54576288 EC50 = 2511.89 nM T11241 C78NBU 54576289 EC50 = 3162.28 nM T11241 CU2Q1F 54576290 EC50 > 3162.28 nM T11241 CVA4I0 54576291 EC50 > 3162.28 nM T11241 C1BQ9K 54576499 EC50 > 3162.28 nM T11241 C4P8DY 54576501 EC50 > 3162.28 nM T11241 CSAV94 54576503 EC50 > 3162.28 nM T11241 CTUN47 54576721 EC50 = 2511.89 nM T11241 C61UKW 54579593 EC50 > 10000 nM T11241 C5M2PI 54580603 IC50 > 20000 nM T11241 CWNO65 54582607 IC50 = 5400 nM T11241 CI20JA 54756906 EC50 > 31622.78 nM T11241 CCG08B 54756907 EC50 > 100000 nM T11241 CK50BF 54756908 EC50 = 6309.57 nM T11241 CILG27 54758399 EC50 = 15848.93 nM T11241 CU62DN 54764919 EC50 > 25000 nM T11241 CHLD32 56834955 EC50 = 2500 nM T11241 CA80UC 56835064 EC50 = 8200 nM T11241 CDN71L 56835182 EC50 = 390 nM T11241 C7HYC3 56948659 EC50 = 630 nM T11241 C64ORS 56951563 EC50 > 25000 nM T11241 CBIH06 56954024 IC50 > 10000 nM T11241 CF2Q9V 56955980 EC50 = 559 nM T11241 C0I9ED 56955982 EC50 = 339 nM T11241 C1LAY2 57335019 EC50 > 2500 nM T11241 CW9QP5 57390104 EC50 > 25000 nM T11241 CM36YP 57390142 EC50 > 25000 nM T11241 CN6LF0 57390143 EC50 > 25000 nM T11241 C8A1WC 57390144 EC50 = 7420 nM T11241 C5PX7M 57390794 EC50 > 25000 nM T11241 CW6VG3 57390795 EC50 > 2500 nM T11241 C4EF3Z 57391457 EC50 = 12000 nM T11241 C3O4YQ 57391821 EC50 = 14000 nM T11241 CT27YQ 57391849 EC50 = 4500 nM T11241 CV7ZY6 57391886 EC50 > 25000 nM T11241 CHMJ97 57391887 EC50 > 25000 nM T11241 CK3X6Y 57391920 EC50 = 1500 nM T11241 CO0CG8 57391921 EC50 = 2500 nM T11241 C2QK1U 57392608 EC50 > 2500 nM T11241 CE0K1G 57392609 EC50 > 25000 nM T11241 CWSR47 57392652 EC50 > 2500 nM T11241 C9B2VK 57393585 EC50 = 11000 nM T11241 CO7A0R 57393586 EC50 > 20000 nM T11241 C0MAT8 57393649 EC50 = 2500 nM T11241 CZT94U 57394329 EC50 = 5560 nM T11241 COJI42 57394406 EC50 > 25000 nM T11241 C4F0IJ 57394951 EC50 = 2000 nM T11241 CU0Z7A 57394952 EC50 = 3000 nM T11241 C5WPX0 57395262 EC50 = 2900 nM T11241 CLM47H 57395264 EC50 = 11000 nM T11241 CB5SI2 57395297 EC50 = 13000 nM T11241 CD1H8X 57395369 EC50 = 2680 nM T11241 CR16YK 57395370 EC50 = 2500 nM T11241 CSG64Z 57395371 EC50 = 2500 nM T11241 CGTY01 57395372 EC50 = 2500 nM T11241 CP56XE 57395373 EC50 = 2500 nM T11241 CZS2J6 57395374 EC50 = 2500 nM T11241 CY5H6S 57396084 EC50 = 1130 nM T11241 CFR73W 57396172 EC50 = 1560 nM T11241 CN98GO 57396699 EC50 = 4600 nM T11241 C8EUA6 57397066 EC50 = 15000 nM T11241 C9MDA7 57397196 EC50 = 900 nM T11241 C9HB5I 57397896 EC50 > 25000 nM T11241 C57RHP 57397897 EC50 = 1440 nM T11241 C3Q8JD 57397984 EC50 > 25000 nM T11241 C6NIS0 57398468 EC50 = 800 nM T11241 C4RPA5 57398469 EC50 > 20000 nM T11241 CR39MB 57398470 EC50 > 20000 nM T11241 CE90LI 57398471 EC50 > 20000 nM T11241 CUPB85 57398603 EC50 > 20000 nM T11241 CJ8LF5 57398802 EC50 = 5000 nM T11241 CD2H4N 57398845 EC50 = 10000 nM T11241 CH2C9P 57398870 EC50 > 25000 nM T11241 CZPO40 57398897 EC50 = 2500 nM T11241 CY98KJ 57399545 EC50 > 2500 nM T11241 CLH87C 57399546 EC50 = 834 nM T11241 CJVQ54 57399579 EC50 > 2500 nM T11241 C3HWU8 57400134 EC50 > 20000 nM T11241 CX2R7O 57400135 EC50 > 20000 nM T11241 C0EH7G 57400136 EC50 > 20000 nM T11241 CVDZ56 57400137 EC50 > 20000 nM T11241 C4A5EH 57400476 EC50 = 22000 nM T11241 CPB4E0 57400520 EC50 > 20000 nM T11241 C93FBE 57400521 EC50 = 6000 nM T11241 CBE5U1 57400584 EC50 > 25000 nM T11241 CFS52K 57400585 EC50 = 2040 nM T11241 CLGZ16 57400586 EC50 = 2500 nM T11241 CXC10U 57400587 EC50 = 2500 nM T11241 CQRU15 57400588 EC50 = 2500 nM T11241 CM8S5O 57401335 EC50 > 2500 nM T11241 C08KNY 57401336 EC50 > 2500 nM T11241 C57BKF 57402280 EC50 = 20800 nM T11241 C5PVG3 57402282 EC50 = 9450 nM T11241 C39PIE 57402284 EC50 = 29300 nM T11241 CBP4S0 57402328 EC50 > 20000 nM T11241 C86CHT 57402358 EC50 = 2060 nM T11241 C5C7JK 57402390 EC50 > 25000 nM T11241 CHO08Y 57402391 EC50 = 2500 nM T11241 CUZB73 57402392 EC50 = 2500 nM T11241 CEH9D3 57403052 EC50 > 25000 nM T11241 CI6J3E 57403053 EC50 > 25000 nM T11241 C6S0XI 57404009 EC50 = 3900 nM T11241 CGE71H 57404012 EC50 > 30000 nM T11241 CR7AU1 57404343 EC50 > 10000 nM T11241 CO8JI5 57404344 EC50 = 501.19 nM T11241 CT9UR5 57404356 EC50 > 10000 nM T11241 C0F5NL 57437353 EC50 = 141 nM T11241 CN49YH 57437389 EC50 = 242 nM T11241 C1QY9C 57505797 EC50 > 31622.78 nM T11241 CDH87C 57505996 EC50 = 31622.78 nM T11241 C3T2KX 57508868 EC50 = 599 nM T11241 CLF0Q9 57522810 EC50 > 10000 nM T11241 C6X2YS 57522811 EC50 > 10000 nM T11241 C52LBR 57522812 EC50 = 2511.89 nM T11241 CN0JL5 57522815 EC50 > 3162.28 nM T11241 CAZ1C6 57522939 EC50 > 3162.28 nM T11241 C6K0OG 57522940 EC50 > 3162.28 nM T11241 CVS1Y9 57522941 EC50 > 10000 nM T11241 C0A1JE 57554662 IC50 > 10000 nM T11241 CLG2V4 57554674 IC50 = 3 nM T11241 C3UX5B 57570459 EC50 = 1600 nM T11241 C7V4JG 57570461 EC50 = 4300 nM T11241 CBF40Z 57570463 EC50 = 1900 nM T11241 CGA79V 57570467 EC50 = 2500 nM T11241 CYW65N 57570476 EC50 = 3200 nM T11241 CYB43R 57570486 EC50 = 1300 nM T11241 C3AD7V 57570487 EC50 = 3000 nM T11241 CJLX28 57570497 EC50 = 5900 nM T11241 CA9CY8 57570498 EC50 = 1500 nM T11241 CZ19YS 57570503 EC50 = 4000 nM T11241 COE91B 57699087 Ki = 4880 nM T11241 C5YS7U 58329611 EC50 > 10000 nM T11241 C30BKS 58390822 EC50 = 720000 nM T11241 CMN68P 58390859 EC50 = 300 nM T11241 C86MRL 58390878 EC50 = 485 nM T11241 CR07UT 58390929 EC50 = 950 nM T11241 CD9SZ5 58390949 EC50 = 4550 nM T11241 C7T0LA 58537167 EC50 > 31 nM T11241 CHU24M 58537193 EC50 = 9200 nM T11241 CZ6R5C 58537228 EC50 = 1300 nM T11241 C4IXQ6 58725140 EC50 > 3000 nM T11241 CM71ZT 58907531 IC50 = 10000 nM T11241 CCJ2B4 58907649 IC50 = 1050 nM T11241 CD6EH2 58907658 IC50 = 10000 nM T11241 CO26CZ 59146063 EC50 > 10000 nM T11241 C74YXS 59146106 EC50 > 10000 nM T11241 C38MAI 59202018 EC50 = 590 nM T11241 CY2M9Z 59202022 EC50 = 1860 nM T11241 C8FZ4S 59384310 EC50 > 3000 nM T11241 CQ52OA 59384375 EC50 > 3000 nM T11241 C3D4EZ 59451753 IC50 > 10000 nM T11241 C1CYE5 59451764 IC50 > 10000 nM T11241 CU83BX 59451813 IC50 > 10000 nM T11241 CB9S0P 59451832 IC50 > 10000 nM T11241 CR62AY 59451867 IC50 > 10000 nM T11241 CCAI45 59451870 IC50 > 10000 nM T11241 C2QZ8N 59495631 Ki = 1040 nM T11241 CJA5S6 59548622 EC50 > 31622.78 nM T11241 C8J6GQ 59593534 EC50 = 5210 nM T11241 CE37MO 59982944 EC50 = 2200 nM T11241 C4MZP6 60150588 EC50 > 20000 nM T11241 C1C8SV 60150616 EC50 > 20000 nM T11241 C07EBJ 66561414 EC50 > 3162.28 nM T11241 C6WM1N 66636736 EC50 = 1253 nM T11241 CPON94 66636757 EC50 = 1150 nM T11241 CF59YL 66636847 EC50 = 247 nM T11241 C7YA0P 66655198 EC50 = 1258.93 nM T11241 CMT3L8 66655210 EC50 = 3981.07 nM T11241 C1M4BX 66655282 EC50 > 10000 nM T11241 CD09QP 66655362 EC50 = 1584.89 nM T11241 CD2I5L 66655520 EC50 > 31622.78 nM T11241 CTX2M1 66655578 EC50 > 10000 nM T11241 CASW54 66655584 EC50 > 1000 nM T11241 CN83CO 66655586 EC50 = 1000 nM T11241 CJG3A2 66655632 EC50 > 10000 nM T11241 CI5KQ1 66655655 EC50 > 10000 nM T11241 CSVZ95 66655679 EC50 > 10000 nM T11241 CRGW91 66655753 EC50 > 10000 nM T11241 C9PGA0 66655774 EC50 > 10000 nM T11241 C7WVE9 66655956 EC50 > 10000 nM T11241 CZS20N 66655962 EC50 > 10000 nM T11241 C6UGD4 66655998 EC50 > 10000 nM T11241 CQ0U7L 66656025 EC50 > 10000 nM T11241 CKO1L6 66656274 EC50 > 10000 nM T11241 CZS9C7 66829256 EC50 = 660 nM T11241 C5E0VD 66829275 EC50 = 45 nM T11241 CGI61O 66829279 EC50 = 150 nM T11241 C4XNF6 66829308 EC50 = 120 nM T11241 C5UTG1 66829311 EC50 = 145 nM T11241 CW9UH3 66829334 EC50 = 20 nM T11241 C5XDU9 66852776 EC50 > 30000 nM T11241 C8Q9HN 66853439 EC50 > 30000 nM T11241 CCBH03 66853698 EC50 > 10000 nM T11241 CG69FE 66923349 EC50 > 3000 nM T11241 CD9BG6 66931911 EC50 = 560 nM T11241 CY25VM 66955367 EC50 = 2100 nM T11241 C8X7CG 66955472 EC50 = 3500 nM T11241 CHZG64 67009121 IC50 > 10000 nM T11241 CF1LH2 67193564 EC50 > 30000 nM T11241 CGOE75 67193675 EC50 > 30000 nM T11241 C19JMK 67193896 EC50 > 30000 nM T11241 C3QCF7 67195432 EC50 > 30000 nM T11241 CN2K6J 67195504 EC50 = 6800 nM T11241 C1CR8J 67195758 EC50 > 30000 nM T11241 CNO54F 67196129 EC50 > 30000 nM T11241 CZ3HJ7 67196477 EC50 > 30000 nM T11241 CVRG24 67197502 EC50 > 30000 nM T11241 C6AZY0 67249162 EC50 > 10000 nM T11241 CX6SF2 67250226 EC50 > 10000 nM T11241 CP0K7H 67266022 EC50 = 1400 nM T11241 CCJ3R5 67284085 EC50 > 31622.78 nM T11241 CT0SQ6 67284109 EC50 > 31622.78 nM T11241 CA8W5X 67284479 EC50 > 19952.62 nM T11241 C8SMB3 67285906 EC50 > 31622.78 nM T11241 CW3JD2 67351486 EC50 = 5270 nM T11241 C0FH4B 67414717 EC50 = 407 nM T11241 CMI48F 67415695 EC50 > 10000 nM T11241 CHFX15 67416434 EC50 = 4200 nM T11241 CVK91L 68192087 EC50 > 3000 nM T11241 CS0GZ3 68446124 EC50 = 1584.89 nM T11241 C0H4RL 68547259 EC50 = 27 nM T11241 CMG53F 68553624 EC50 = 47 nM T11241 C2KI7M 68555865 EC50 = 33 nM T11241 C4Q3NF 68762699 EC50 = 29 nM T11241 CD98MX 68763522 EC50 = 318 nM T11241 CT3PC6 69143493 EC50 > 10000 nM T11241 CXZ2A1 69143673 EC50 = 2590 nM T11241 CS2W7J 69144360 EC50 = 4630 nM T11241 C8RG2L 69144892 EC50 > 10000 nM T11241 CV4OD5 69144893 EC50 > 10000 nM T11241 CF76YV 69144915 EC50 = 1610 nM T11241 CQ9N2R 69145858 EC50 > 10000 nM T11241 CY09OV 69263869 EC50 = 2880 nM T11241 CCFQ57 70681006 EC50 > 10000 nM T11241 CQ27UW 70681007 EC50 > 10000 nM T11241 C6PG3U 70681008 EC50 > 10000 nM T11241 C6D9LM 70681009 EC50 > 10000 nM T11241 CY28VU 70681258 EC50 > 10000 nM T11241 C9UD6M 70681384 EC50 = 400 nM T11241 CH42VZ 70681385 EC50 > 20000 nM T11241 CMZ6I4 70681674 EC50 > 10000 nM T11241 CX26ST 70681687 EC50 = 199.53 nM T11241 CRQO04 70681688 EC50 = 501.19 nM T11241 CC3SF4 70681689 EC50 = 1995.26 nM T11241 C30MIN 70681812 EC50 > 25000 nM T11241 C8CX6G 70681813 EC50 = 5600 nM T11241 CKS42M 70681814 EC50 > 25000 nM T11241 CALO30 70681815 EC50 = 1600 nM T11241 C7IE8O 70683136 EC50 > 10000 nM T11241 C9CND8 70683137 EC50 > 10000 nM T11241 CTH29P 70683346 EC50 > 10000 nM T11241 CEJ51S 70683347 EC50 > 10000 nM T11241 CIOV12 70683348 EC50 > 10000 nM T11241 CR03ZG 70683349 EC50 > 10000 nM T11241 C8BSP9 70683465 EC50 > 20000 nM T11241 CZFR46 70683478 EC50 > 20000 nM T11241 CQ29EW 70683479 EC50 > 20000 nM T11241 CQ2O3C 70683480 EC50 > 20000 nM T11241 CH81TY 70683793 EC50 > 10000 nM T11241 CHM21Y 70683794 EC50 > 10000 nM T11241 CR19FO 70683922 EC50 > 25000 nM T11241 CK1Z3U 70685208 EC50 > 10000 nM T11241 CLV2B8 70685209 EC50 > 10000 nM T11241 CX8HF7 70685210 EC50 > 3162.28 nM T11241 CG0B8I 70685211 EC50 > 10000 nM T11241 CQS7I1 70685573 EC50 > 20000 nM T11241 CXBU72 70685582 EC50 > 20000 nM T11241 C51SBP 70685583 EC50 > 20000 nM T11241 C0ZIF9 70685933 EC50 > 10000 nM T11241 CZ19QH 70685934 EC50 > 10000 nM T11241 C7MZQ0 70685935 EC50 > 10000 nM T11241 C8L0XD 70685939 EC50 = 501.19 nM T11241 CXU38H 70686050 EC50 > 25000 nM T11241 C2ILY4 70686051 EC50 = 1100 nM T11241 CNI10K 70686052 EC50 = 940 nM T11241 CZY89T 70686053 EC50 > 25000 nM T11241 CL31YJ 70687367 EC50 > 10000 nM T11241 CLK95G 70687368 EC50 > 10000 nM T11241 CN8Z6V 70687369 EC50 > 3162.28 nM T11241 C6JM8Q 70687592 EC50 > 10000 nM T11241 CF1CE4 70687715 EC50 > 20000 nM T11241 C02SFN 70687728 EC50 > 20000 nM T11241 CA7RO8 70687729 EC50 > 20000 nM T11241 C2XU1Y 70687730 EC50 > 20000 nM T11241 CCQ97S 70688066 EC50 > 10000 nM T11241 COCF48 70688067 EC50 > 10000 nM T11241 CP3UG2 70688177 EC50 = 1300 nM T11241 CQ0ZN8 70688528 EC50 > 10000 nM T11241 C8Q6YJ 70689430 EC50 > 10000 nM T11241 CGYX75 70689431 EC50 > 10000 nM T11241 CGPI21 70689432 EC50 > 10000 nM T11241 CW51BD 70689433 EC50 = 2511.89 nM T11241 CTI8V1 70689434 EC50 > 10000 nM T11241 CC8E7V 70689644 EC50 > 10000 nM T11241 CLHV45 70689764 EC50 > 20000 nM T11241 CG65PK 70689765 EC50 > 20000 nM T11241 CCB9W1 70689781 EC50 > 20000 nM T11241 CNS91B 70689782 EC50 > 20000 nM T11241 CO8TR9 70690085 EC50 > 10000 nM T11241 CJ5KM4 70690096 EC50 = 125.89 nM T11241 CIMG07 70691539 EC50 > 10000 nM T11241 C13XWD 70691540 EC50 > 10000 nM T11241 CY78XU 70691541 EC50 > 10000 nM T11241 CD9HK6 70691922 EC50 > 20000 nM T11241 CRV82N 70692232 EC50 > 10000 nM T11241 CO5G0D 70692233 EC50 > 10000 nM T11241 CI01GS 70692234 EC50 > 10000 nM T11241 CPIX90 70692235 EC50 > 10000 nM T11241 CAJ78G 70692236 EC50 > 10000 nM T11241 C1C0DO 70692237 EC50 > 10000 nM T11241 C5PT2V 70692238 EC50 > 10000 nM T11241 CVOW40 70692256 EC50 = 1000 nM T11241 C1FIS9 70692257 EC50 = 1995.26 nM T11241 C9Z5LN 70692258 EC50 = 1995.26 nM T11241 C92JOF 70692370 EC50 > 25000 nM T11241 C7UNV3 70692732 EC50 > 10000 nM T11241 CYAS67 70693630 EC50 > 10000 nM T11241 CIG81N 70693631 EC50 > 10000 nM T11241 C9V3GW 70693632 EC50 > 10000 nM T11241 CO0A1Z 70693633 EC50 > 10000 nM T11241 C0OA7T 70693634 EC50 > 10000 nM T11241 C3NC8P 70693635 EC50 > 3162.28 nM T11241 CT7S1Z 70693636 EC50 > 3162.28 nM T11241 CJSX34 70693847 EC50 > 10000 nM T11241 COP46G 70693848 EC50 > 10000 nM T11241 CT5J1F 70693975 EC50 > 20000 nM T11241 C7DFY6 70693976 EC50 > 20000 nM T11241 CD6I5X 70694325 EC50 = 251.19 nM T11241 CT12OX 70694326 EC50 = 1258.93 nM T11241 CXIB79 70694327 EC50 = 1000 nM T11241 CB7CT3 70694328 EC50 = 794.33 nM T11241 C76HLN 70694426 EC50 > 25000 nM T11241 C8PK5N 70694427 EC50 > 25000 nM T11241 CDQ83S 70695740 EC50 > 10000 nM T11241 CQBH21 70695741 EC50 > 10000 nM T11241 CBUZ83 70695742 EC50 > 10000 nM T11241 CFL2H8 70695743 EC50 = 1584.89 nM T11241 C3EAN4 70695958 EC50 > 10000 nM T11241 CXJ78C 70696095 EC50 > 20000 nM T11241 C9HWE1 70696096 EC50 > 20000 nM T11241 CW0LC8 70696401 EC50 > 10000 nM T11241 CA20YS 70696402 EC50 > 10000 nM T11241 C6WO5Y 70696411 EC50 = 1995.26 nM T11241 CCF0R3 70696493 EC50 > 25000 nM T11241 CR4V0T 71450073 IC50 = 802 nM T11241 CMQ9J5 71487023 EC50 > 10000 nM T11241 CQV01F 71487029 EC50 > 10000 nM T11241 C16KJX 71540398 IC50 > 10000 nM T11241 CB87GJ 71540499 IC50 > 10000 nM T11241 CK39OJ 72546270 EC50 = 8070 nM T11241 C85WKP 72793738 EC50 > 10000 nM T11241 C1SC2N 72793739 EC50 > 10000 nM T11241 CSJ7L9 72793740 EC50 > 10000 nM T11241 CWIK42 72793741 EC50 > 10000 nM T11241 CI0N5T 72793759 EC50 > 10000 nM T11241 CNBK82 72793774 EC50 > 10000 nM T11241 C38DCV 72793775 EC50 > 10000 nM T11241 COHM70 72793788 EC50 = 5030 nM T11241 CEG7U8 72793789 EC50 = 1070 nM T11241 CASW13 72793790 EC50 = 348 nM T11241 CHO28L 72793791 EC50 = 870 nM T11241 C1Y6MK 72793810 EC50 = 19.9 nM T11241 CJ56PQ 72793811 EC50 = 65.3 nM T11241 C3YQ2R 72793820 EC50 > 10000 nM T11241 C9D5RT 72793821 EC50 > 10000 nM T11241 CP2M4D 72793822 EC50 = 7 nM T11241 C9K8YM 72793828 EC50 = 110 nM T11241 CJ48WM 73333750 EC50 = 1273 nM T11241 CHMD43 73774584 EC50 = 383 nM T11241 C6G3YC 76310852 EC50 = 24 nM T11241 COQY72 76310992 EC50 = 24 nM T11241 C2DB3P 76310993 EC50 = 5240 nM T11241 CW48DP 76310994 EC50 = 2630 nM T11241 C2H9FK 76311230 EC50 = 1790 nM T11241 C3TGY9 76311231 EC50 = 1000 nM T11241 CL6ZD0 76311232 EC50 = 21 nM T11241 CA3L2S 76314472 EC50 = 83 nM T11241 CC9W0M 76314473 EC50 = 819 nM T11241 C56OGS 76314474 EC50 = 8.9 nM T11241 CEN46O 76314475 EC50 > 10000 nM T11241 C8MFO0 76314621 EC50 = 3.6 nM T11241 C68NUF 76314622 EC50 = 5 nM T11241 C39OGP 76314623 EC50 = 868 nM T11241 C04AUW 76314624 EC50 = 866 nM T11241 C7AI9H 76314625 EC50 = 25 nM T11241 CHYG50 76314626 EC50 > 10000 nM T11241 CB9L0F 76318055 EC50 = 26 nM T11241 CQ6E1G 76318056 EC50 = 11 nM T11241 C2TL1H 76318057 EC50 = 3830 nM T11241 CWC1G2 76318058 EC50 = 172 nM T11241 C4O8RP 76318194 EC50 > 10000 nM T11241 CYJ3Z8 76318195 EC50 = 9950 nM T11241 CH9B3U 76318196 EC50 = 3730 nM T11241 CF7X8W 76318197 EC50 = 1230 nM T11241 CR6H1D 76318198 EC50 = 617 nM T11241 CY2CW5 76318199 EC50 = 1770 nM T11241 CA1I7G 76318200 EC50 = 2900 nM T11241 C6UDP4 76318445 EC50 = 349 nM T11241 C69WSQ 76318446 EC50 = 391 nM T11241 C08KVJ 76321769 EC50 = 172 nM T11241 C1CZ0H 76321770 EC50 = 15 nM T11241 CLB13F 76321771 EC50 > 10000 nM T11241 CKR7X3 76321772 EC50 = 11 nM T11241 CJ69NG 76321773 EC50 = 3910 nM T11241 C87GMQ 76321895 EC50 = 1340 nM T11241 CB0N9L 76321896 EC50 = 24 nM T11241 CGC85U 76321897 EC50 = 5740 nM T11241 C2V5AL 76322116 EC50 = 3.72 nM T11241 CA9V2U 76322117 EC50 = 184 nM T11241 C7UL9Q 76322118 EC50 = 2100 nM T11241 CVP6Y8 76322119 EC50 = 302 nM T11241 CKUS39 76322127 EC50 = 1711 nM T11241 C3NK2P 76322128 EC50 = 2197 nM T11241 CQ17WJ 76325392 EC50 = 62 nM T11241 C4VG0E 76325528 EC50 = 2.4 nM T11241 C90FKU 76325529 EC50 = 25 nM T11241 CXA1J3 76325530 EC50 = 429 nM T11241 C3SDU8 76325531 EC50 = 1120 nM T11241 C9ZQ3K 76325533 EC50 = 106 nM T11241 CGLB78 76325739 EC50 = 1000 nM T11241 C54XGU 76325748 EC50 = 1141 nM T11241 C8IX9H 76325749 EC50 > 5000 nM T11241 CN14OE 76328931 EC50 = 25 nM T11241 CE5D9I 76329073 EC50 = 258 nM T11241 CMG6Q7 76329074 EC50 > 10000 nM T11241 CQ5HF1 76329075 EC50 = 700 nM T11241 CX4OA0 76329076 EC50 = 3080 nM T11241 CNH32U 76329077 EC50 > 10000 nM T11241 CO9QF7 76329310 EC50 > 5000 nM T11241 CF84JV 76329311 EC50 = 508 nM T11241 C3EKT6 76329326 EC50 = 225 nM T11241 CYP53V 76329327 EC50 = 1739 nM T11241 CA7GO0 76332613 EC50 > 10000 nM T11241 CI48VM 76332614 EC50 > 10000 nM T11241 CPCU86 76332615 EC50 = 1.2 nM T11241 CE0U5H 76332741 EC50 = 149 nM T11241 CNI13W 76332955 EC50 = 113 nM T11241 CCJ1E9 76332956 EC50 = 204 nM T11241 CP4M6B 76332957 EC50 = 1000 nM T11241 C5ZW4J 76336211 EC50 = 5.8 nM T11241 COB8X9 76336212 EC50 = 15 nM T11241 CNJ13I 76336213 EC50 = 5270 nM T11241 C0XIK8 76336214 EC50 = 25 nM T11241 CFU3C9 76336215 EC50 > 10000 nM T11241 CVM60F 76336361 EC50 = 3940 nM T11241 C1VJZ3 76336362 EC50 = 860 nM T11241 CGTV16 76336363 EC50 = 5960 nM T11241 C0O2NK 76336364 EC50 = 429 nM T11241 COX87F 76336566 EC50 = 1130 nM T11241 C1EZ9S 76336567 EC50 = 1000 nM T11241 CB5NI0 76336568 EC50 = 130 nM T11241 C42TIC 76336569 EC50 = 674 nM T11241 C9IKU5 78321974 EC50 > 1000 nM T11241 CK4S8A 86646444 EC50 > 10000 nM T11241 CL3Y8J 89484779 IC50 > 800 nM T11241 CI1WF3 89710483 EC50 > 10000 nM T11241 C2G1HE 89710485 EC50 > 10000 nM T11241 CJ6RC9 89710536 EC50 = 1584.89 nM T11241 CGE95T 89710694 EC50 > 10000 nM T11241 CLP73T 89710808 EC50 > 10000 nM T11241 CR0LX1 89711073 EC50 > 10000 nM T11241 C2D4SQ 89713031 EC50 > 1000 nM T11241 C0TQK5 89713056 EC50 > 10000 nM T11241 CQ3PK4 90308914 IC50 > 800 nM T11241 C89FXZ 90309040 IC50 > 800 nM T11241 CYSQ05 90309100 IC50 > 800 nM T11241 CL74JM 90309142 IC50 > 10000 nM T11241 CY3ZT1 90309524 IC50 > 800 nM T11241 CY7K8V 91758813 EC50 > 10000 nM T11241 C3XVO1 101863648 IC50 = 4900 nM T11241 C51VMH 118707012 EC50 = 200 nM T11241 C5K8VH 118707193 EC50 = 180 nM T11241 CX1UP2 118707194 EC50 > 20000 nM T11241 CEI4M5 118707195 EC50 = 60 nM T11241 CKR17A 118707196 EC50 = 220 nM T11241 CA0K5C 118707197 EC50 = 12000 nM T11241 C9SQ5X 118707198 EC50 = 340 nM T11241 CL1EJ7 118707199 EC50 > 20000 nM T11241 C9C0FB 118716137 EC50 > 5000 nM T11241 CQJ87G 118716138 EC50 = 1945 nM T11241 CMJ7B8 118716139 EC50 = 1020 nM T11241 C4D5QX 118716140 EC50 = 1113 nM T11241 CK0C5M 118716141 EC50 = 245 nM T11241 C3C6VG 118716142 EC50 = 569 nM T11241 C6S5FV 118716143 EC50 = 356 nM T11241 CSR50K 118716144 EC50 = 2110 nM T11241 CP6W7I 118716145 EC50 = 416 nM T11241 C3KN6Y 118716146 EC50 = 237 nM T11241 CPR5Y4 118716147 EC50 = 844 nM T11241 CH0P9G 118716148 EC50 = 2973 nM T11241 CA10EJ 118716149 EC50 > 5000 nM T11241 CM14DZ 118716150 EC50 = 869 nM T11241 CG3OD8 118716151 EC50 > 5000 nM T11241 C8XNF6 118716152 EC50 = 899.2 nM T11241 COIL26 118716153 EC50 = 828 nM T11241 C4QBP2 118716154 EC50 = 970 nM T11241 C5JTY2 118716155 EC50 = 1391 nM T11241 CL78NH 118716156 EC50 = 925 nM T11241 CSP01A 118716157 EC50 = 1544 nM T11241 C2WY3I 118716177 EC50 = 1388 nM T11241 CJ2X5A 118716178 EC50 = 3008 nM T11241 C0N6LQ 118716179 EC50 > 5000 nM T11241 CGQ3D4 118716180 EC50 = 1997 nM T11241 CI6J2D 118716181 EC50 = 616 nM T11241 COX9P3 118716182 EC50 = 1219 nM T11241 C79NHT 118716183 EC50 = 1910 nM T11241 CTQO81 118716184 EC50 = 496 nM T11241 C3L2JK 118716185 EC50 = 4689 nM T11241 C0AK1I 118716186 EC50 = 1390 nM T11241 CV2NB9 118716187 EC50 > 5000 nM T11241 C86HJL 118716188 EC50 > 5000 nM T11241 C5T1DG 118716189 EC50 > 5000 nM T11241 CJ0PM8 118716190 EC50 > 5000 nM T11241 CB25DV 118717764 EC50 = 450 nM T11241 CH43DI 118717765 EC50 > 10000 nM T11241 CV8IT1 118717766 EC50 > 10000 nM T11241 C41LOQ 118717769 EC50 > 10000 nM T11241 CP1VA0 118717770 EC50 > 10000 nM T11241 C2HTU4 118717771 EC50 = 4700 nM T11241 CRS38A 118717772 EC50 > 10000 nM T11241 CJC90W 118717773 EC50 > 10000 nM T11241 CFH74U 118717774 EC50 > 10000 nM T11241 C5NVP7 118717775 EC50 > 10000 nM T11241 CH7OB1 118717776 EC50 > 10000 nM T11241 CPG9M3 118717777 EC50 = 410 nM T11241 CK2L1R 118717778 EC50 = 380 nM T11241 CS62RG 118717779 EC50 > 10000 nM T11241 CHV80J 118717780 EC50 > 10000 nM T11241 C5QG8O 118717781 EC50 > 10000 nM T11241 C3BX4H 118717782 EC50 > 10000 nM T11241 CIKX78 118717783 EC50 > 10000 nM T11241 CT85QI 118717784 EC50 > 10000 nM T11241 C69IKB 118717785 EC50 > 10000 nM T11241 C6XA2I 118717786 EC50 > 10000 nM T11241 C9GN1O 118717787 EC50 > 10000 nM T11241 CQ8E5P 118717788 EC50 > 10000 nM T11241 C5JVO1 118717789 EC50 > 10000 nM T11241 CW7Y8V 118717790 EC50 > 10000 nM T11241 CLXR38 118717791 EC50 > 10000 nM T11241 CW5XJ2 118717792 EC50 > 10000 nM T11241 CA6N4E 118717793 EC50 > 10000 nM T11241 CS4V1Q 118717794 EC50 > 10000 nM T11241 CV83BZ 118717795 EC50 = 940 nM T11241 C6Y0VB 118723864 EC50 = 3981.07 nM T11241 CK23TG 118724202 EC50 > 31622.78 nM T11241 CFL73Q 118724203 EC50 > 31622.78 nM T11241 CNI96W 118728428 IC50 > 25000 nM T11241 C3O6KB 118728429 IC50 > 25000 nM T11241 C4U3DG 118728430 IC50 > 800 nM T11241 C8U0GE 118728431 IC50 > 800 nM T11241 C72NCP 118728432 IC50 > 10000 nM T11241 C2YHT8 118728433 IC50 > 25000 nM T11241 C4M3YA 118728434 IC50 > 25000 nM T11241 CH23UV 124171442 EC50 > 10000 nM T11241 C9VT4Z 124171444 EC50 > 10000 nM T11241 CX8VT2 124171447 EC50 > 10000 nM T11241 CONE63 124171453 EC50 > 10000 nM T11241 CE8C9A 124171498 EC50 > 10000 nM T11241 C9U4QR 124221654 EC50 > 100000 nM T11241 CE6YZ3 127025658 EC50 > 31622.78 nM T11241 CP2OX6 127027154 EC50 = 19952.62 nM T11241 CL5IF7 127028461 EC50 > 31622.78 nM T11241 C95FHV 127028462 EC50 > 31622.78 nM T11241 C1LJ2E 127028463 EC50 > 31622.78 nM T11241 CDQ8X2 127028464 EC50 > 31622.78 nM T11241 C63BMS 127028465 EC50 > 31622.78 nM T11241 C01GPK 127029098 EC50 > 31622.78 nM T11241 CIM27T 127029099 EC50 > 31622.78 nM T11241 CPT32H 127029100 EC50 > 31622.78 nM T11241 C0WPV4 127029101 EC50 > 31622.78 nM T11241 CQT30N 127029102 EC50 > 31622.78 nM T11241 C7QMK2 127032587 EC50 = 1058 nM T11241 C6W7TO 127032588 EC50 > 10000 nM T11241 CREP02 127032589 EC50 = 484 nM T11241 CI51JP 127034581 EC50 > 10000 nM T11241 CL70FK 127037694 IC50 = 40 nM T11241 CQ37LX 127037695 IC50 = 23 nM T11241 CM54QV 127037696 IC50 = 5290 nM T11241 CD52GS 127041987 IC50 = 197 nM T11241 CG90DH 127045708 EC50 = 5100 nM T11241 CT2FY0 127045962 EC50 = 4400 nM T11241 CN8Y5X 127045963 EC50 = 370 nM T11241 C0WDZ1 127046095 EC50 = 2900 nM T11241 C1HW3J 127046096 EC50 = 1200 nM T11241 CXM68P 127046097 EC50 > 10000 nM T11241 CNVH82 127046130 EC50 = 6300 nM T11241 C1FPU6 127046179 EC50 = 2300 nM T11241 C9QXJ5 127046183 EC50 = 1600 nM T11241 C7XSZ6 127046184 EC50 = 95 nM T11241 C91DCL 127046185 EC50 = 110 nM T11241 C6PU3Y 127046323 EC50 = 5500 nM T11241 CDKY27 127046324 EC50 > 10000 nM T11241 CX38TU 127046325 EC50 = 210 nM T11241 CE2O1K 127046399 EC50 = 800 nM T11241 C63EGK 127046400 EC50 = 180 nM T11241 CG06MF 127046456 EC50 = 2100 nM T11241 C6CZ1K 127046548 EC50 = 71 nM T11241 C09FWP 127046549 EC50 = 140 nM T11241 CHQ87M 127046550 EC50 = 17 nM T11241 CG90HA 127046551 EC50 = 38 nM T11241 CPV3A5 127046566 EC50 = 1500 nM T11241 CLS7H0 127046567 EC50 = 930 nM T11241 CR25DJ 127046568 EC50 = 1400 nM T11241 CVRA82 127046640 EC50 > 10000 nM T11241 CT1U5D 127046641 EC50 > 10000 nM T11241 CL5PG6 127046741 EC50 = 190 nM T11241 C83BTN 127046742 EC50 = 55 nM T11241 CPB61O 127046743 EC50 = 50 nM T11241 CH6W9G 127046863 EC50 > 10000 nM T11241 CA40VG 127046864 EC50 > 10000 nM T11241 C3RCI0 127046865 EC50 > 10000 nM T11241 CNX35J 127046866 EC50 = 4600 nM T11241 C1M3IE 127046992 EC50 = 3100 nM T11241 C05PXK 127047020 EC50 = 22 nM T11241 C76SEA 127047083 EC50 = 210 nM T11241 C7WS0V 127047084 EC50 = 920 nM T11241 C63NVZ 127047144 EC50 > 10000 nM T11241 C9J1HQ 127047145 EC50 > 10000 nM T11241 C5CSZ1 127047225 EC50 > 10000 nM T11241 C1PFQ4 127047226 EC50 > 10000 nM T11241 CY5O0B 127047690 EC50 > 10000 nM T11241 CCEF35 127047778 EC50 > 10000 nM T11241 C4KL3G 127047779 EC50 = 9000 nM T11241 C0Y3WZ 127047780 EC50 = 4300 nM T11241 CB43PM 127047986 EC50 > 10000 nM T11241 CHC04K 127048099 EC50 = 1700 nM T11241 CP91CD 127048100 EC50 > 10000 nM T11241 CYDJ81 127048101 EC50 > 10000 nM T11241 C7L2PZ 127048102 EC50 = 8100 nM T11241 CM9L1X 127048104 EC50 > 10000 nM T11241 CO0I8C 127048141 EC50 = 870 nM T11241 C25KAZ 127048142 EC50 = 560 nM T11241 CDZ3C4 127048143 EC50 = 1500 nM T11241 CR47MS 127048144 EC50 > 10000 nM T11241 CUE0N7 134130169 EC50 > 100000 nM T11241 C3NC1O 134130546 EC50 > 100000 nM T11241 CJH4K9 134130548 EC50 > 100000 nM T11241 C6JB4Z 134130695 EC50 > 100000 nM T11241 C6V4DA 134130884 EC50 > 100000 nM T11241 CNVC46 134131381 EC50 > 100000 nM T11241 CRB05V 134319250 EC50 > 3000 nM T11241 C2JQ7P 134319251 EC50 > 3000 nM T11241 C2KHY7 134319262 EC50 > 3000 nM T11241 CSK4I8 134319263 EC50 > 3000 nM T11241 CUH3P6 134319264 EC50 > 3000 nM T11241 C8ZX0N 134319265 EC50 > 3000 nM T11241 CRS09O 134319702 EC50 = 190 nM T11241 CZ8MH2 136053659 EC50 > 31622.78 nM T11241 C2CHL4 137638716 IC50 = 1200 nM T11241 C81HEI 137644547 Ki = 2200 nM T11241 C42VXM 137646436 EC50 > 31000 nM T11241 CAJY69 137651211 IC50 = 100 nM T11241 C25TZL 137655932 IC50 = 280 nM T11241 CH2AN7 137660780 IC50 > 10000 nM T11241 CHRG61 145964044 EC50 > 10000 nM T11241 C0ZM4R 145966230 IC50 > 1000 nM T11241 CR8Q4L 145969830 EC50 > 10000 nM T11241 CN8IE0 145975394 EC50 = 1995.26 nM T11241 C6JW8K 145976329 IC50 > 1000 nM T11241 C7MI9V 145978086 EC50 > 10000 nM T11241 CRF7V0 155317229 IC50 > 1000 nM T11241 CX76PB 155317261 IC50 > 1000 nM T11241 CW10AC 155317265 IC50 > 1000 nM T11241 C43CXP 155317276 IC50 > 1000 nM T11241 CLG86C 155317279 IC50 > 1000 nM T11241 CC17FU 155513062 EC50 > 31000 nM T11241 CD73QT 155522973 EC50 = 2100 nM T11241 CI3BA5 155527137 EC50 = 3800 nM T11241 C9I7SA 155528529 EC50 = 14000 nM T11241 CL0E5D 155534250 EC50 = 1100 nM T11241 CE4W7D 155537600 EC50 = 10000 nM T11241 C37AGW 155538268 EC50 = 14000 nM T11241 C78VOU 155542034 EC50 = 7400 nM T11241 CI4X9B 155543631 EC50 = 4800 nM T11241 CH28SZ 155550350 EC50 = 2500 nM T11241 CPY85W 16215109 EC50 > 1000 nM T11241 CZSI05 44438257 EC50 > 1000 nM T11241 CWKU57 44438259 EC50 > 1000 nM T11241 CT3AX1 44438261 EC50 > 1000 nM T11241 D00VHN 46905530 IC50 = 6.3 nM T11241 D02LTS 59393720 IC50 > 10000 nM T11241 D04IAF 11452022 EC50 = 0.134 nM T11241 D04XCB 10149595 IC50 > 10000 nM T11241 D05EDD 11588811 EC50 = 450 nM T11241 D05KEE 10904818 EC50 = 6.31 nM T11241 D06DYN 9908268 EC50 = 0.1 nM T11241 D06GFH 11545181 Ki = 300 nM T11241 D06XMB 44394220 IC50 = 27 nM T11241 D07EAB 10215259 IC50 = 2100 nM T11241 D08VLT 10125714 IC50 = 6600 nM T11241 D0D5QS 11725751 IC50 = 2.7 nM T11241 D0LO4T 10287034 IC50 = 18 nM T11241 D0N0BN 44394248 IC50 = 370 nM T11241 D0P1TY 44344193 IC50 = 3.6 nM T11241 D0P2AZ 10149721 IC50 = 4900 nM T11241 D0ZU0O 4077460 EC50 > 25000 nM T33902 D00QET 5281040 Ki = 6540 nM T33902 D05EJG 6305 IC50 > 30000 nM T33902 D08QIP 4887 Ki = 4060 nM T33902 D0R1RS 3715 IC50 = 28800 nM T33902 D0S9MU 5078 IC50 > 30000 nM T33902 D0O6AQ 6450546 Ki = 1630 nM T33902 CMZ76T 88264 EC50 = 1140 nM T33902 CK2DH4 169313 EC50 > 30000 nM T33902 CC1V0H 446916 EC50 = 331 nM T33902 C7WXA8 963505 EC50 > 30000 nM T33902 C4DF0S 4052279 EC50 = 3720 nM T33902 C6P7VU 5311303 IC50 = 508 nM T33902 C25RID 9796971 EC50 > 30000 nM T33902 CT73IB 10260031 IC50 = 0.7 nM T33902 CPS7J5 10566103 EC50 > 30000 nM T33902 COK96Y 10671020 IC50 = 582 nM T33902 CO2VH9 11433866 EC50 = 0.036 nM T33902 CEH9S8 13792576 EC50 > 30000 nM T33902 CE9DP2 14783466 EC50 > 30000 nM T33902 CILP95 14783467 EC50 = 30000 nM T33902 C76UDK 15747648 EC50 >= 10000 nM T33902 C19IOR 15747649 EC50 >= 10000 nM T33902 C43PDX 15747650 EC50 = 7410 nM T33902 CFZ5M6 15747651 IC50 = 8400 nM T33902 CQ9L5R 15747652 EC50 > 100000 nM T33902 CW4L3E 15747657 EC50 = 270 nM T33902 CK08FE 15747661 EC50 > 30000 nM T33902 C90LGF 22163898 EC50 = 2240 nM T33902 C6S9WH 22163902 EC50 = 45500 nM T33902 C5ZL2X 23279502 IC50 = 112 nM T33902 CL9Z0M 44296063 EC50 > 30000 nM T33902 CZ6J0D 44755067 EC50 = 1.4 nM T33902 CUNX18 46222214 EC50 = 11 nM T33902 C3JX9N 46222216 EC50 = 1.7 nM T33902 CP8FZ1 49797716 EC50 = 945 nM T33902 CASU41 71280744 EC50 = 5440 nM T33902 CJA36G 71280754 EC50 > 100000 nM T33902 CJK21G 71280760 EC50 = 4830 nM T33902 C6P4RK 71280839 EC50 > 100000 nM T33902 C06SCJ 71280847 EC50 = 4020 nM T33902 CRL7M6 71280862 EC50 = 731 nM T33902 C2LVW0 71280863 EC50 = 3010 nM T33902 CRG0Z7 71280865 EC50 = 4980 nM T33902 CCX70G 71280866 EC50 = 202 nM T33902 CYO96U 71280879 EC50 = 715 nM T33902 C9Z4LE 71280882 EC50 = 52000 nM T33902 C9FEP0 71280939 EC50 = 4790 nM T33902 CL9D2P 71280970 EC50 = 7900 nM T33902 CK13JC 71281042 EC50 > 100000 nM T33902 CRF3S4 71281161 EC50 = 4090 nM T33902 CC6SP7 71281217 EC50 = 9550 nM T33902 CV5PL8 71281224 EC50 = 14400 nM T33902 CJ9Z1N 71281286 EC50 = 4130 nM T33902 C5RFB3 71281465 EC50 = 15100 nM T33902 COAJ50 76311173 EC50 = 17100 nM T33902 CP64BC 76314777 EC50 = 36800 nM T33902 CHQ63V 96412014 EC50 = 1680 nM T33902 CJ5O7T 131858496 EC50 > 30000 nM T33902 C9S6UV 145964032 EC50 = 117 nM T33902 CN9V3P 145964575 EC50 = 423 nM T33902 CY1LC3 145965055 EC50 > 100000 nM T33902 CF19IO 145965176 EC50 > 100000 nM T33902 CXN9I8 145965484 EC50 = 3680 nM T33902 C3Z9SD 145965649 EC50 > 10000 nM T33902 CE28XN 145965896 EC50 > 30000 nM T33902 CC1WJ7 145968969 EC50 > 30000 nM T33902 CX2P3J 145969377 EC50 > 30000 nM T33902 CUOG29 145971655 EC50 = 27.9 nM T33902 CZE31S 145971828 EC50 = 67 nM T33902 C8Q9JF 145971888 EC50 > 10000 nM T33902 C36WRU 145971906 EC50 = 624 nM T33902 CZJ0G2 145972277 EC50 > 30000 nM T33902 C12ETR 145972331 EC50 = 1470 nM T33902 C4RL5Z 145976960 EC50 >= 10000 nM T33902 CGL4F7 145977144 EC50 = 115 nM T33902 CPS91R 145978078 EC50 = 32.1 nM T33902 C7X6FU 145978218 EC50 = 103 nM T33902 D02VPC 1826 IC50 > 30000 nM T80024 CRS87L 118732224 IC50 = 4100 nM T80024 CSD16Y 118732229 IC50 = 3560 nM T80024 C9E3GH 134137378 IC50 = 1190 nM T80024 CP8I7R 137634541 IC50 = 320 nM T80024 C7SU2J 155519745 IC50 = 130 nM T80024 CQ4JP9 155540392 IC50 = 260 nM T68290 D00TLP 24873435 IC50 = 800 nM T68290 D0V3YT 10324367 IC50 = 120 nM T68290 D0X9CH 3010818 IC50 = 300 nM T68290 D0J6AU 10152654 IC50 = 45 nM T68290 D0HM5J 118253852 IC50 > 20000 nM T68290 D01LNG 10201696 IC50 = 2900 nM T68290 D0T5PH 6918602 Ki = 1.6 nM T68290 CV8A4D 163098 IC50 = 400 nM T68290 C8OHY9 254021 IC50 = 6000 nM T68290 CI0DG1 764318 IC50 > 200000 nM T68290 CPA63I 3107941 IC50 > 200000 nM T68290 C6SO2K 3708081 IC50 > 200000 nM T68290 CR2ND4 5287468 Ki = 4 nM T68290 CW6D7Z 5287498 IC50 = 1200 nM T68290 CB6H0T 5287549 Ki = 8.3 nM T68290 CS96RK 5287799 IC50 = 19 nM T68290 CESY50 5288259 IC50 = 5.2 nM T68290 C6YF4B 5288616 IC50 = 150 nM T68290 CFM6E4 5288618 IC50 = 260 nM T68290 C9E1UW 5288633 Ki > 1000 nM T68290 CN3RY0 5289345 Ki = 890 nM T68290 CR68MZ 6323453 Ki = 3800 nM T68290 C1DAZ6 6420159 Ki = 29 nM T68290 C0XQP7 6917747 IC50 > 100000 nM T68290 CN26IL 9547980 Ki = 32 nM T68290 CCZ83F 9808750 Ki < 100 nM T68290 CQ1NG7 9815041 IC50 = 1578 nM T68290 C03AMQ 9822322 IC50 = 23 nM T68290 C9F7PL 9825191 Ki = 1960 nM T68290 C0N4DH 9825355 IC50 = 2000 nM T68290 CK7B2P 9829646 IC50 = 46 nM T68290 CCD9G5 9830736 IC50 = 50 nM T68290 C2IGS5 9831164 IC50 = 13 nM T68290 CN1EH9 9843168 IC50 = 47 nM T68290 CLQ92U 9848147 IC50 = 4600 nM T68290 C2VX4Z 9848148 Ki = 3290 nM T68290 C10QOS 9874384 IC50 = 10 nM T68290 CL4VY9 9874885 Ki = 8100 nM T68290 CO0PD1 9883178 IC50 = 63 nM T68290 C0NM3D 9887557 IC50 = 1.5 nM T68290 CGA91J 9890145 IC50 = 2800 nM T68290 C8P5LN 9891030 Ki = 5600 nM T68290 C8HI1R 9891108 IC50 = 1600 nM T68290 C5L4YE 9893225 IC50 = 0.5 nM T68290 COK50T 9895628 IC50 = 2 nM T68290 C2JCM5 9902742 IC50 = 9000 nM T68290 C5XS2F 9904539 Ki = 620 nM T68290 CALH63 9908450 IC50 = 1340 nM T68290 C7WKG9 9913437 IC50 = 9500 nM T68290 CXD2Y6 9926586 IC50 = 400 nM T68290 CT74FA 9933804 IC50 = 10 nM T68290 C5ZD9R 9943969 IC50 > 1000 nM T68290 CNR6D5 9948720 IC50 = 10 nM T68290 C4WFJ2 9980678 Ki = 188 nM T68290 CBNR45 9980918 IC50 > 1000 nM T68290 CHN80D 9981917 IC50 > 10000 nM T68290 C1F4BA 9984481 IC50 = 1.9 nM T68290 C8RCT2 10002592 IC50 = 5 nM T68290 C7P6JO 10004326 IC50 > 1000 nM T68290 C40APB 10005577 IC50 > 1000 nM T68290 CI96RJ 10008050 IC50 < 0.4 nM T68290 CXY9N8 10024008 IC50 > 1000 nM T68290 CLB5G0 10025017 IC50 = 13 nM T68290 C4NW7I 10026902 IC50 = 800 nM T68290 C0SJY5 10031327 IC50 = 1.5 nM T68290 CJO52T 10046162 IC50 > 1000 nM T68290 CU1EF5 10047111 IC50 = 77 nM T68290 C68HGW 10047261 IC50 = 102 nM T68290 C8F7MU 10047536 IC50 > 1000 nM T68290 CXH45E 10051341 IC50 = 76 nM T68290 C6O8RU 10072812 IC50 = 210 nM T68290 CV29YC 10076076 IC50 = 37 nM T68290 CHA42Q 10097070 IC50 = 9500 nM T68290 C8FPB5 10098917 IC50 = 0.5 nM T68290 CA5N3E 10111943 IC50 = 34 nM T68290 C57JDN 10118049 IC50 = 1.3 nM T68290 CFC3Q8 10120133 IC50 = 530 nM T68290 C87RIK 10120530 IC50 = 72 nM T68290 C6AZ3B 10120903 IC50 = 19000 nM T68290 CR1Z9B 10121038 IC50 = 100 nM T68290 CAMC60 10121688 IC50 = 50 nM T68290 CD87QK 10121801 IC50 = 23 nM T68290 C97NJR 10121949 Ki = 13000 nM T68290 C5OTM3 10121955 IC50 = 21 nM T68290 C2E9OK 10122123 IC50 = 44 nM T68290 C53MDT 10122124 IC50 = 34 nM T68290 CSF93N 10122137 IC50 = 180 nM T68290 C9L2UX 10122216 IC50 = 33 nM T68290 C3VE4T 10122218 IC50 = 220 nM T68290 C7XOA0 10127183 IC50 = 172 nM T68290 CSO96K 10127748 IC50 = 20 nM T68290 CKZ15P 10129236 IC50 = 27 nM T68290 CJ79ZX 10138553 IC50 = 8340 nM T68290 CY6PU1 10143615 Ki = 110 nM T68290 CLID02 10144235 Ki = 45000 nM T68290 CY0XH8 10144986 IC50 = 360 nM T68290 CQ9Z2V 10145669 IC50 = 58 nM T68290 CX69MD 10146027 IC50 = 29 nM T68290 CR71XJ 10146491 IC50 = 27 nM T68290 CQ3YD8 10150891 IC50 = 365 nM T68290 C8DQG0 10154619 IC50 = 922 nM T68290 CO2Z7G 10155296 IC50 > 1000 nM T68290 C9VFI4 10161284 Ki = 13000 nM T68290 C1Q2EX 10164497 Ki = 470 nM T68290 CDX7R4 10164961 IC50 = 3700 nM T68290 C5B1HM 10165557 IC50 = 750 nM T68290 CTJ7R3 10166544 IC50 = 78 nM T68290 CDRE91 10167323 Ki = 20000 nM T68290 CI7OY9 10167456 IC50 = 80 nM T68290 CN0A9X 10167663 IC50 = 10 nM T68290 C6NHP8 10167901 IC50 = 600 nM T68290 CZW7M5 10168197 IC50 = 29 nM T68290 CSUI41 10168223 IC50 = 800 nM T68290 CME0C3 10168439 IC50 = 37 nM T68290 C0Y2RQ 10168654 IC50 = 80 nM T68290 CQ8GN0 10168898 IC50 = 1200 nM T68290 CG2HI9 10168928 IC50 = 130 nM T68290 CU16HJ 10169029 IC50 = 47 nM T68290 CZ1A8U 10173731 IC50 = 153 nM T68290 C5NEX6 10174161 IC50 = 11 nM T68290 C1YR4T 10174359 IC50 = 17 nM T68290 CD4G7F 10179450 IC50 = 24 nM T68290 CTON03 10179451 IC50 = 158 nM T68290 C07GUT 10184761 Ki = 1800 nM T68290 C4M3SG 10186046 IC50 = 110000 nM T68290 CCO7A6 10187105 Ki = 17000 nM T68290 C0SF7U 10187920 IC50 = 160 nM T68290 C15LHK 10188965 IC50 = 38 nM T68290 CO8P7B 10189260 IC50 = 50 nM T68290 C4EUC3 10189472 IC50 = 145 nM T68290 CWVU18 10189565 IC50 = 30 nM T68290 CKZ1A0 10194354 IC50 = 62 nM T68290 CZD7A6 10194447 IC50 = 240 nM T68290 CA2UH4 10194634 IC50 = 449 nM T68290 CQ8YM3 10199981 Ki = 16000 nM T68290 CL9DW3 10200425 IC50 = 1245 nM T68290 CG7E3L 10208282 IC50 = 9500 nM T68290 C9K6IU 10208398 IC50 = 2100 nM T68290 CR0L4W 10210806 IC50 = 95 nM T68290 CS3IP7 10210867 IC50 = 1600 nM T68290 C7XL5J 10210875 IC50 = 50 nM T68290 CC05SY 10210876 IC50 = 27 nM T68290 CVL86X 10211091 IC50 = 195 nM T68290 CC5HG7 10211194 IC50 = 240 nM T68290 C1WL9J 10211340 Ki = 3300 nM T68290 CFX7Z2 10211615 IC50 = 30 nM T68290 C3BXH9 10211620 IC50 = 54 nM T68290 CGI4W0 10211816 IC50 = 50 nM T68290 CEN82K 10211864 IC50 = 16 nM T68290 C1F9SP 10216231 IC50 = 1698 nM T68290 C1Y3QZ 10216510 IC50 = 614 nM T68290 C5GSN6 10216511 IC50 = 278 nM T68290 C17RPY 10230100 IC50 = 1000 nM T68290 CT8K5D 10231379 IC50 = 0.21 nM T68290 C4OZ5K 10231447 IC50 = 520 nM T68290 C7WBU8 10232449 IC50 = 120 nM T68290 CVY65P 10232596 IC50 = 120 nM T68290 C7UOX6 10232786 IC50 = 20 nM T68290 C20FGH 10233020 IC50 = 80 nM T68290 C6W9BP 10233130 IC50 = 100 nM T68290 CM7H2R 10233142 IC50 = 170 nM T68290 C6EM9B 10233328 IC50 = 826 nM T68290 CER43X 10233451 IC50 = 18 nM T68290 CPRC34 10233559 IC50 = 18 nM T68290 CZ7TP4 10233786 IC50 = 30 nM T68290 CJBI61 10237771 IC50 = 54 nM T68290 CFI43Z 10238903 IC50 = 154 nM T68290 CORW86 10247897 IC50 = 840 nM T68290 CEQ21I 10249499 IC50 > 1000 nM T68290 C6A8NV 10252643 Ki = 180 nM T68290 CP13MQ 10252805 IC50 = 5.5 nM T68290 CO5EZ1 10257915 Ki = 4000 nM T68290 C56PLQ 10258908 Ki = 39000 nM T68290 C9SOH2 10271564 IC50 = 652 nM T68290 CBHO04 10272927 IC50 > 1000 nM T68290 C6A5CZ 10281649 IC50 = 120 nM T68290 CPQ42Z 10282468 IC50 = 77 nM T68290 CE5BP1 10282652 IC50 = 140 nM T68290 C49OTB 10282988 IC50 = 32 nM T68290 CESR87 10283088 IC50 = 130 nM T68290 CGJ97C 10284032 IC50 = 39 nM T68290 CKX0R7 10287617 IC50 = 121 nM T68290 CUW38E 10288162 IC50 = 189 nM T68290 CX23AL 10288163 IC50 = 249 nM T68290 CY7DQ2 10288811 IC50 = 34 nM T68290 CV9LB1 10302710 IC50 = 720 nM T68290 CUQ2R3 10303526 IC50 = 3700 nM T68290 CV5S7B 10303657 IC50 = 19000 nM T68290 CS3DV6 10303703 IC50 = 100 nM T68290 CZR02J 10303878 Ki = 10000 nM T68290 CK80OJ 10304088 IC50 = 120 nM T68290 CA7IV3 10304215 IC50 = 25 nM T68290 C3NJ2U 10304660 IC50 = 60 nM T68290 CS3Y6X 10304727 IC50 = 23 nM T68290 C4GE9V 10305094 IC50 = 140 nM T68290 CLQ0A4 10305142 IC50 = 130 nM T68290 CPT49O 10310362 IC50 = 607 nM T68290 C9DN6G 10325113 IC50 < 0.4 nM T68290 C59ZDR 10337631 IC50 = 920 nM T68290 C2GLK6 10346121 IC50 = 48 nM T68290 CDX2C8 10367993 IC50 > 1000 nM T68290 CYF98Z 10368089 IC50 = 1900 nM T68290 CX7S8A 10392779 IC50 = 0.58 nM T68290 CF7O6A 10409137 IC50 = 2.8 nM T68290 C41JUO 10414118 IC50 = 4.9 nM T68290 CDVZ19 10431266 Ki = 950 nM T68290 C8DTH3 10436731 IC50 = 937 nM T68290 CN18SE 10456222 Ki = 0.26 nM T68290 C06QJW 10457653 IC50 = 330 nM T68290 C5M7BL 10471316 IC50 = 460 nM T68290 CXD68E 10473874 IC50 = 68 nM T68290 C9D7XO 10478741 IC50 = 930 nM T68290 C32MAD 10482525 IC50 < 0.4 nM T68290 C1MX2S 10499322 Ki = 1100 nM T68290 CHTL13 10507714 Ki = 90 nM T68290 C25HQJ 10522795 Ki > 1000 nM T68290 C0UBF5 10524384 Ki = 480 nM T68290 CR54HQ 10569603 Ki > 10000 nM T68290 C8U1RQ 10593841 Ki = 310 nM T68290 CJ7U3O 10668284 IC50 > 10000 nM T68290 C9V5EX 10673009 Ki = 20 nM T68290 CRL23A 10674588 Ki = 910 nM T68290 C9PY4N 10690022 Ki = 530 nM T68290 CKO6L0 10698950 Ki = 8 nM T68290 C9AIY1 10793962 Ki = 51 nM T68290 C9XI7T 10804795 IC50 > 10000 nM T68290 CQ08YK 10807774 Ki > 1000 nM T68290 CHC3F0 10817683 Ki = 97 nM T68290 CZ4V0F 10832380 Ki > 10000 nM T68290 CA3SY1 10858935 IC50 = 97000 nM T68290 CW7AI1 10860703 IC50 = 107000 nM T68290 CBWJ85 10862359 IC50 = 3931 nM T68290 CNVG58 10875013 IC50 = 190 nM T68290 C85CYF 10884634 IC50 = 9 nM T68290 C7ZNC2 10892596 IC50 = 226 nM T68290 CZK49P 10893343 IC50 = 1257 nM T68290 CYF7Z3 10893503 IC50 = 17 nM T68290 CE85IB 10895386 IC50 = 9 nM T68290 CNX10K 10895470 IC50 = 5 nM T68290 C5PF2M 10896077 IC50 = 8 nM T68290 CWXN58 10902758 Ki = 46000 nM T68290 CBJ1I7 10902914 IC50 > 10000 nM T68290 CA30HS 10905508 IC50 = 6597 nM T68290 C8D2FC 10906131 IC50 = 12 nM T68290 C5X6NA 10924832 IC50 > 10000 nM T68290 C6TPH0 10927935 IC50 = 173 nM T68290 C3YFK8 10938614 IC50 = 19 nM T68290 CZG37Y 10938664 IC50 > 10000 nM T68290 C7YR3J 10938777 IC50 = 21 nM T68290 CA72YH 10949332 IC50 = 48 nM T68290 CKG53T 10960024 IC50 = 41 nM T68290 CL7W4P 10960628 IC50 = 1550 nM T68290 CW1L5K 10960899 IC50 = 7200 nM T68290 CR0P8J 10971179 IC50 > 10000 nM T68290 CK9E8W 10972182 IC50 > 10000 nM T68290 C6ZOI1 10979734 IC50 = 8039 nM T68290 CG67WO 10982531 IC50 = 84 nM T68290 CN4LS6 10990120 IC50 = 142 nM T68290 C4PNO3 10992343 IC50 = 6000 nM T68290 CA3NG9 10993428 IC50 = 2310 nM T68290 CM9Z5T 11012257 IC50 > 10000 nM T68290 CV0MO9 11013354 IC50 = 134000 nM T68290 C5XHI0 11014664 IC50 = 9422 nM T68290 C5PFZ9 11024844 IC50 > 28000 nM T68290 CY72BF 11034349 IC50 > 10000 nM T68290 C4C3OT 11046559 IC50 = 51 nM T68290 CY0LF2 11058796 IC50 = 8 nM T68290 CVC74W 11059260 IC50 = 56 nM T68290 C56CUP 11059525 IC50 = 7 nM T68290 CHN48V 11069367 IC50 = 9 nM T68290 CY3V4J 11080121 IC50 = 88 nM T68290 C0PSR8 11081485 IC50 = 1298 nM T68290 C5WY1H 11082075 IC50 = 1200 nM T68290 C27DYK 11098017 IC50 = 124 nM T68290 CL0Z2O 11120472 IC50 = 114 nM T68290 CQ4L0T 11122768 IC50 = 5700 nM T68290 CQK6U4 11144121 IC50 = 4000 nM T68290 CDR7A6 11155973 Ki = 1 nM T68290 C8EAL0 11156785 Ki = 11 nM T68290 C9SN1Q 11157631 Ki = 5 nM T68290 CH41OF 11157632 Ki = 69 nM T68290 C61AIQ 11168385 Ki = 60 nM T68290 CAI94Q 11168613 Ki = 27 nM T68290 C2VJG7 11178623 Ki = 19 nM T68290 CJW65I 11178915 Ki < 100 nM T68290 CMDU74 11180007 Ki = 24 nM T68290 C9ZNL4 11191320 Ki > 4500 nM T68290 CS90MB 11191512 Ki = 12 nM T68290 C2H4GP 11200735 Ki = 98 nM T68290 CTCX89 11203484 Ki = 105 nM T68290 C17UIX 11203679 IC50 = 50 nM T68290 C7SOL0 11224927 Ki = 93 nM T68290 CM8ZV1 11225780 Ki = 28 nM T68290 CLC2X1 11226457 Ki = 28 nM T68290 C0JO5R 11238059 Ki = 21 nM T68290 C3T1LM 11238468 Ki = 71 nM T68290 CQ32YR 11238775 IC50 = 14000 nM T68290 C5VY1E 11247716 Ki = 43 nM T68290 CLA6J3 11249688 Ki = 88 nM T68290 CRXU26 11250282 Ki = 200 nM T68290 CHK9N2 11261516 Ki = 62 nM T68290 C8F2ZN 11269453 IC50 > 1000 nM T68290 CIFQ06 11273375 Ki = 7 nM T68290 C15XUE 11283547 Ki = 25 nM T68290 CCH6N4 11283555 IC50 = 265 nM T68290 CM86BP 11294094 Ki = 173 nM T68290 CFU50G 11294227 Ki = 26 nM T68290 CV86IB 11295906 Ki = 68 nM T68290 CZX89I 11305296 Ki = 197 nM T68290 CR2T5B 11305867 Ki = 6 nM T68290 CU6Z0F 11306593 Ki = 9.1 nM T68290 CEC0A2 11316876 Ki = 222 nM T68290 CDYL91 11327594 Ki = 1721 nM T68290 CP5MI6 11329727 Ki = 95 nM T68290 CD70PA 11341599 Ki = 11 nM T68290 C5X1VW 11351327 IC50 = 0.4 nM T68290 CFJ70U 11353015 Ki = 15 nM T68290 C9W0TB 11375856 Ki = 134 nM T68290 C7NQX3 11375955 Ki = 11 nM T68290 CH4I3T 11375956 IC50 = 71 nM T68290 C34DFQ 11376188 Ki = 27 nM T68290 CAL7B2 11376611 Ki = 43 nM T68290 COV1F4 11387157 Ki = 261 nM T68290 CEW0F3 11387421 Ki = 34 nM T68290 C3DQL2 11396020 Ki = 1368 nM T68290 C4QM7I 11396148 Ki = 94 nM T68290 CER2V8 11397519 Ki = 43 nM T68290 C4ZLU9 11397590 Ki = 194 nM T68290 C7RFC5 11398171 Ki = 16 nM T68290 CI3HK2 11409407 Ki = 15 nM T68290 CO4Y3H 11410560 Ki = 616 nM T68290 CU4P8A 11418931 Ki = 196 nM T68290 C56SXA 11419952 Ki = 47 nM T68290 CGD1K4 11421700 Ki = 8 nM T68290 CILJ37 11431699 Ki = 31 nM T68290 CM2VQ6 11431993 Ki = 151 nM T68290 C19YRB 11432272 Ki = 38 nM T68290 C72PFO 11432501 Ki = 3 nM T68290 C65ASH 11432773 Ki = 1590 nM T68290 CQRB45 11433280 Ki = 18 nM T68290 CQIP48 11439739 IC50 = 200 nM T68290 CME0C5 11443502 Ki = 434 nM T68290 CH9ZA7 11443990 Ki = 26 nM T68290 C1AT2Z 11453155 IC50 = 0.6 nM T68290 CL53MS 11456165 Ki = 730 nM T68290 CME32S 11456379 Ki = 405 nM T68290 C0O8MK 11464526 IC50 = 210 nM T68290 C5N3BV 11466327 Ki = 12 nM T68290 CV43WB 11466677 Ki = 13 nM T68290 CM59AQ 11466845 Ki = 12 nM T68290 CL1D2Z 11471738 IC50 = 158 nM T68290 C0ZK5I 11477975 Ki = 14 nM T68290 C9U0YI 11478637 Ki = 37 nM T68290 CBC8U6 11490230 Ki = 21 nM T68290 C94SZC 11493500 Ki = 860 nM T68290 CZLF20 11494632 Ki = 440 nM T68290 CR2M4H 11494672 Ki = 190 nM T68290 CM41QW 11494775 Ki = 180 nM T68290 CT8S4U 11496335 Ki = 7900 nM T68290 C5CL9A 11496988 Ki = 6 nM T68290 CC92RV 11501571 IC50 = 4800 nM T68290 CFI8L5 11502586 IC50 = 18 nM T68290 CK5JM6 11503223 Ki = 4900 nM T68290 CY4A7V 11504785 Ki = 27 nM T68290 C3Q7BE 11504819 Ki = 300 nM T68290 CCH09G 11507712 Ki > 150000 nM T68290 CHI9N5 11512144 Ki = 42000 nM T68290 CF20TJ 11514361 Ki > 100000 nM T68290 C23DKS 11516307 IC50 = 23 nM T68290 CDA9F5 11517167 Ki = 110000 nM T68290 C6B5UF 11520360 IC50 = 41000 nM T68290 C87YFV 11523212 Ki = 83 nM T68290 C6D2VI 11525733 Ki = 8700 nM T68290 CW4ED1 11532268 IC50 = 2 nM T68290 CQ69XF 11533114 Ki = 26000 nM T68290 C2BT3L 11533910 Ki = 17000 nM T68290 CQ6UC2 11537070 Ki = 770 nM T68290 CY0AV1 11544076 Ki = 760 nM T68290 C6XK8V 11547772 Ki = 21000 nM T68290 C65NQY 11550481 Ki = 28000 nM T68290 CG57TI 11551229 Ki = 13600 nM T68290 CYO67B 11551502 Ki = 2100 nM T68290 C3BTN5 11556651 IC50 = 36000 nM T68290 CXTQ39 11558838 Ki = 3500 nM T68290 CF9DE7 11561418 Ki = 102000 nM T68290 CA61ZJ 11562424 Ki = 7900 nM T68290 CKH13D 11562461 Ki = 16000 nM T68290 CTN57Q 11562607 Ki = 3900 nM T68290 CMH1V5 11563622 IC50 = 48000 nM T68290 CB3W8O 11565199 Ki = 490 nM T68290 CPY84F 11569750 Ki = 9100 nM T68290 CW1O0M 11569883 Ki = 6200 nM T68290 C8T5DM 11570453 IC50 = 21000 nM T68290 C1TV6S 11580329 Ki = 14000 nM T68290 C9YNX2 11581727 Ki = 340 nM T68290 CB1L7I 11583999 IC50 = 170000 nM T68290 C73VCU 11584899 Ki = 8.9 nM T68290 CJG6T3 11585276 Ki = 3.1 nM T68290 CER65Q 11588182 Ki = 240 nM T68290 CUX70T 11588744 Ki = 4000 nM T68290 C2Y6JE 11590993 Ki = 13000 nM T68290 CLV84W 11594784 Ki = 34000 nM T68290 C1QO2C 11598043 IC50 = 2 nM T68290 CR9VG2 11599767 IC50 > 150000 nM T68290 CQZ5T4 11602113 Ki = 31000 nM T68290 C7X0QE 11602978 Ki = 0.9 nM T68290 CT8XH2 11603305 Ki > 100000 nM T68290 C1NV2U 11605163 Ki = 68000 nM T68290 CM4OS2 11606272 Ki = 5.7 nM T68290 C98KMP 11612451 Ki = 250 nM T68290 CZU5E4 11613136 Ki = 19000 nM T68290 CW0T9J 11613973 IC50 = 77000 nM T68290 CK0AN9 11616537 Ki = 15000 nM T68290 C7W8JG 11616689 Ki > 100000 nM T68290 CE8WO5 11618337 Ki = 5700 nM T68290 CTL1P3 11618795 Ki = 2500 nM T68290 CH21OU 11623464 Ki = 2800 nM T68290 CQ7KD1 11623853 Ki = 150 nM T68290 C9LBF3 11628054 Ki = 350 nM T68290 CUS5Q4 11630803 Ki = 6500 nM T68290 C3XO5G 11631355 Ki = 2200 nM T68290 C70VTY 11631953 Ki = 6200 nM T68290 C98QKS 11635243 Ki = 42 nM T68290 CLUA24 11636269 IC50 = 12000 nM T68290 CLMY50 11641509 Ki = 30000 nM T68290 CNH8C7 11646581 Ki = 270 nM T68290 C2XHN1 11646851 Ki = 15000 nM T68290 CILB73 11649751 Ki = 3 nM T68290 C8NZX4 11651881 Ki = 650 nM T68290 C2PM1X 11652420 Ki > 50000 nM T68290 CJRN14 11655672 Ki = 20000 nM T68290 C5ZOM0 11656060 IC50 = 7 nM T68290 CO76PW 11659287 Ki = 1700 nM T68290 C0Q7AH 11662896 Ki = 12000 nM T68290 CXU57J 11663056 IC50 = 6.6 nM T68290 C4YFI9 11663730 IC50 < 1 nM T68290 C0D7NS 11663810 Ki = 6400 nM T68290 CYR86V 11664755 IC50 = 35000 nM T68290 CSD3H5 11666846 Ki = 1900 nM T68290 C5SJ9K 11669355 IC50 > 10000 nM T68290 C13TGX 11671560 Ki = 5500 nM T68290 CKH3O7 11673861 Ki > 100000 nM T68290 CT0OZ8 11673881 Ki = 860 nM T68290 C1BGL5 11677886 Ki = 20000 nM T68290 C23ZVP 11678241 Ki = 41 nM T68290 C27LJY 11678922 Ki = 15.6 nM T68290 CDNH37 11680631 Ki > 150000 nM T68290 C1Q2OT 11682028 Ki = 8800 nM T68290 C6Q8KO 11682184 Ki = 1400 nM T68290 CNB67S 11684874 Ki = 33000 nM T68290 CL4XB1 11685284 Ki = 92 nM T68290 C53OYX 11692372 Ki = 5.8 nM T68290 C38REW 11695166 Ki > 150000 nM T68290 C6F1GI 11695261 Ki = 44 nM T68290 CJB3E9 11695584 Ki = 35000 nM T68290 C0OC5V 11696208 Ki = 1900 nM T68290 C5H2GL 11696621 Ki = 610 nM T68290 CHP6U3 11699298 Ki = 3200 nM T68290 C7QIP8 11699507 Ki = 8.3 nM T68290 C45DTR 11702249 Ki = 25 nM T68290 CRTS62 11703216 Ki = 300 nM T68290 C5UEI7 11703527 IC50 = 47 nM T68290 C9X6PV 11703830 Ki = 9.2 nM T68290 C0Y5XV 11705688 Ki = 42000 nM T68290 CRZ6T0 11709547 Ki = 590 nM T68290 CT4QY5 11710096 Ki = 1300 nM T68290 C5FZ1J 11710873 IC50 = 16 nM T68290 C5ME9N 11716536 Ki = 270 nM T68290 C26RZY 11717535 Ki = 10000 nM T68290 CJ1L4F 11729761 IC50 = 6 nM T68290 C5JMK8 11731802 IC50 = 11000 nM T68290 CPL53T 11732127 IC50 = 76000 nM T68290 CMX6H5 11732856 IC50 = 9 nM T68290 CDS4P0 11743922 Ki = 46 nM T68290 C0SV2T 11753412 Ki = 5 nM T68290 CY63BP 11761693 IC50 = 470 nM T68290 C8D7BS 11771234 Ki > 10 nM T68290 CSO1F8 11783702 IC50 > 339000 nM T68290 CT5B1S 11784942 Ki = 2130 nM T68290 CLSM45 11809509 IC50 = 1400 nM T68290 CZ7PO1 11810830 IC50 = 130 nM T68290 C71CHA 11811466 IC50 > 13000 nM T68290 CDJH89 11811557 IC50 = 1695 nM T68290 CU5B0A 11823521 IC50 = 82 nM T68290 CGP3Z2 11823960 IC50 = 56 nM T68290 CZ1YB3 11824245 IC50 > 10000 nM T68290 CT38BL 11826257 IC50 = 9 nM T68290 CRXO59 11857300 IC50 = 0.4 nM T68290 CDOG76 11857302 IC50 = 0.7 nM T68290 C5NR3L 11962098 IC50 = 47 nM T68290 C3QN1E 11983275 Ki = 350 nM T68290 C31MCN 13186896 IC50 > 100000 nM T68290 C4JQR9 14060550 Ki > 1000000 nM T68290 COP0K2 14308232 Ki > 100000 nM T68290 C9WC6M 14655218 Ki = 510 nM T68290 CM7H4S 15283376 Ki = 292000 nM T68290 CCGS52 15547237 IC50 = 58 nM T68290 CLGV32 15547238 IC50 = 207 nM T68290 CI8QZ5 15567852 Ki > 1000000 nM T68290 CVO9K6 15858812 IC50 = 430 nM T68290 CHC31Q 15985697 IC50 = 217 nM T68290 C9LW6H 15985754 IC50 = 38 nM T68290 CQ5F9T 16045426 IC50 = 30 nM T68290 CL38RU 16046125 Ki = 19 nM T68290 CQ2N8D 16046128 Ki = 658 nM T68290 C08XJK 16090559 Ki = 1200 nM T68290 CTIV96 16090560 Ki = 420 nM T68290 C2QWA9 16090561 Ki = 200 nM T68290 CJBT92 16090562 IC50 = 10 nM T68290 CU6KB8 16090563 IC50 = 9 nM T68290 CZ9J6G 16108888 IC50 = 0.7 nM T68290 C3KMJ0 16108889 IC50 = 2.3 nM T68290 CM7DA6 16108890 IC50 = 1.6 nM T68290 C0M1KY 16108891 IC50 = 0.9 nM T68290 C63XFT 16108892 IC50 = 3.1 nM T68290 C0LJ8Y 16108893 IC50 = 2.5 nM T68290 C7IQ0W 16108894 IC50 = 0.9 nM T68290 CPN5S2 16108895 IC50 = 2.6 nM T68290 CJ98LN 16108900 IC50 = 0.13 nM T68290 CYT2X8 16108901 IC50 = 0.23 nM T68290 CJRB12 16108902 IC50 = 0.48 nM T68290 C0QAC5 16108903 IC50 > 10 nM T68290 CT65ZO 16108904 IC50 = 1.8 nM T68290 CHKR18 16108905 IC50 = 10 nM T68290 CZI27Q 16108906 IC50 = 0.51 nM T68290 C6D4FQ 16655063 IC50 = 11 nM T68290 C5FUL9 16661369 IC50 = 41082 nM T68290 CUTI57 16661526 IC50 = 76938 nM T68290 C26JIW 16661682 IC50 = 66656 nM T68290 C8QD4E 16662142 IC50 = 25 nM T68290 C6XPN4 16664855 IC50 = 16 nM T68290 C8XLP2 16720100 Ki = 9.6 nM T68290 C4P8ZV 16720327 Ki = 48.7 nM T68290 CI0WO4 17747162 IC50 = 10000 nM T68290 CCPD37 17747164 IC50 = 32 nM T68290 CB7M2X 17747165 IC50 = 35 nM T68290 C9QRT6 17747166 IC50 = 27 nM T68290 CKA87T 17945762 IC50 = 41 nM T68290 CTQM93 17968180 IC50 > 1000 nM T68290 CH4TC1 17968209 IC50 > 1000 nM T68290 C0Q1ML 17968234 IC50 = 460 nM T68290 C0JBH9 18395047 IC50 > 2500 nM T68290 C2XTI9 18395048 IC50 > 2500 nM T68290 C7WD4Z 18628647 IC50 = 1365 nM T68290 CR7B9L 18628679 IC50 = 3343 nM T68290 CHA0S3 18628693 IC50 = 1421 nM T68290 CU3NM9 18628717 IC50 = 6623 nM T68290 C71IFZ 18628739 IC50 > 10000 nM T68290 CUSD12 18628799 IC50 = 609 nM T68290 C34QUK 21309371 IC50 > 2500 nM T68290 CTR87E 22293600 IC50 = 110 nM T68290 CK74TL 22293626 IC50 = 100 nM T68290 COS7Y0 22293642 IC50 = 140 nM T68290 CQ7RT2 22293646 IC50 = 310 nM T68290 CP6VM4 22293649 IC50 = 88 nM T68290 CLD60H 22293656 IC50 = 120 nM T68290 C5H1DR 22293657 IC50 = 68 nM T68290 CJA5G0 22293663 IC50 = 140 nM T68290 CP51WI 22293672 IC50 = 230 nM T68290 CCV37T 22293696 IC50 = 65 nM T68290 CK0QF6 22293697 IC50 = 130 nM T68290 C5A8OE 22293700 IC50 = 150 nM T68290 C04RVW 22293715 IC50 = 1800 nM T68290 CBQN59 22293722 IC50 = 33 nM T68290 CQ7I9S 22293725 IC50 = 50 nM T68290 CK3FH9 22293729 IC50 = 800 nM T68290 C0R3PW 22293758 IC50 = 60 nM T68290 CH6M9Q 22293759 IC50 = 210 nM T68290 CL5G4R 22293772 IC50 = 133 nM T68290 CJ5P6Y 22293788 IC50 = 130 nM T68290 C20MGL 22293806 IC50 = 163 nM T68290 CI86WH 22293808 IC50 = 500 nM T68290 CWB1A0 22293812 IC50 = 110 nM T68290 CQ8FY0 22293823 IC50 = 60 nM T68290 C2KY9R 22293828 IC50 = 120 nM T68290 C0QIZ4 22293838 IC50 = 460 nM T68290 CGQ9P8 22293858 IC50 = 1925 nM T68290 CN5AZ3 22293860 IC50 = 100 nM T68290 CU3XR0 22293870 IC50 = 48 nM T68290 C5G9LB 22293890 IC50 = 90 nM T68290 C4OWK9 22293895 IC50 = 90 nM T68290 CS9LH6 22293909 IC50 = 48 nM T68290 C0XJ4N 22311998 IC50 = 100 nM T68290 C2KBL6 22972497 IC50 = 1427 nM T68290 CD5R3V 22972573 IC50 = 1991 nM T68290 CI57HS 22988111 Ki = 1780 nM T68290 CKW6Q8 23626706 IC50 = 2.5 nM T68290 CZ8DI1 23643986 Ki = 5.5 nM T68290 C0QVL2 23644739 Ki = 107 nM T68290 CM1C8V 23644740 Ki = 23 nM T68290 CM5TI6 23644741 Ki = 149 nM T68290 CMQ72V 23644742 Ki = 12600 nM T68290 CZPF48 23648277 IC50 = 10 nM T68290 CHU59C 23648278 IC50 = 80 nM T68290 CA74XT 23648279 IC50 = 2173 nM T68290 C2I6RW 23648280 IC50 = 10 nM T68290 CCJ8M5 23648281 IC50 = 729 nM T68290 C9C0HK 23648282 IC50 = 6.4 nM T68290 CC50JD 23648283 IC50 = 2.5 nM T68290 CS1VW7 23648284 IC50 = 0.5 nM T68290 CUQH43 23648285 IC50 = 0.3 nM T68290 CM52JD 23648286 IC50 = 0.3 nM T68290 CE09VM 23648287 IC50 = 1.8 nM T68290 C1FRI4 23648288 IC50 = 627 nM T68290 C9RNB7 23648289 IC50 = 0.4 nM T68290 C4J5MD 23648290 IC50 = 0.3 nM T68290 CY20DH 23648291 IC50 = 0.2 nM T68290 CF7O3H 23648292 IC50 = 5 nM T68290 CKI1W5 23648293 IC50 = 1.3 nM T68290 CN5S3K 23648294 IC50 = 0.2 nM T68290 CTB69E 23648295 IC50 = 0.2 nM T68290 C31XJH 23648296 IC50 = 1 nM T68290 C5ECI8 23648297 IC50 = 6183 nM T68290 CB7T3I 23648298 IC50 = 1308 nM T68290 CVF2M6 23648299 IC50 = 36 nM T68290 CRZ56K 23648300 IC50 = 303 nM T68290 CQ1C8H 23648301 IC50 = 282 nM T68290 CQFD10 23648302 IC50 = 196 nM T68290 CFR23Q 23648303 IC50 = 265 nM T68290 C0FBS2 23648304 IC50 = 220 nM T68290 C67AYX 23648305 IC50 = 254 nM T68290 CN6R9M 23648306 IC50 = 436 nM T68290 C85PXH 23648308 IC50 = 653 nM T68290 CVH82R 23648309 IC50 = 188 nM T68290 COZK65 23648310 Ki = 62 nM T68290 CCF89E 23648311 Ki = 46 nM T68290 CS4NV6 23648312 Ki = 23 nM T68290 CC9S7T 23648313 Ki = 9.7 nM T68290 CCTK94 23648314 Ki = 38 nM T68290 CG29HR 23648315 Ki = 285 nM T68290 CY35VT 23648316 Ki = 29 nM T68290 CTX79K 23648317 Ki = 16 nM T68290 C8T5FW 23648318 Ki = 33 nM T68290 C02UQZ 23648319 Ki = 35 nM T68290 C1QVI4 23648320 Ki = 27 nM T68290 CP4SY0 23648321 Ki = 19 nM T68290 C9C7JR 23648322 Ki = 66 nM T68290 CTY4J2 23648323 Ki = 123 nM T68290 CGJ96H 23648326 Ki > 20000 nM T68290 CSI84Q 23648327 Ki > 65000 nM T68290 C2PD6A 23648328 Ki = 16 nM T68290 C37FRY 23648329 Ki = 29 nM T68290 C4KU8Q 23648330 Ki = 34 nM T68290 C09TQZ 23648331 Ki > 20000 nM T68290 CM0AG6 23648332 Ki = 5 nM T68290 C8DJZ7 23648333 Ki = 9.4 nM T68290 CVH46G 23648334 Ki = 2.9 nM T68290 C1IRW9 23648335 Ki = 7.4 nM T68290 CWG7T3 23648336 Ki = 8 nM T68290 CZN75B 23648337 Ki = 17 nM T68290 CLZX16 23648338 Ki = 4 nM T68290 C5UDE3 23648339 Ki = 26 nM T68290 C7V6EY 23648340 Ki = 2 nM T68290 CRK1M0 23648341 Ki = 107 nM T68290 C34VFB 23648342 Ki = 49 nM T68290 CQUD83 23648343 Ki = 34 nM T68290 C32GYK 23648344 Ki = 7.1 nM T68290 CHQ82B 23648345 Ki = 132 nM T68290 CH0XM8 23648346 Ki = 104 nM T68290 C8ZT0W 23648347 Ki = 458 nM T68290 C5T6WQ 23648348 Ki = 563 nM T68290 CKE2C0 23648349 Ki = 230 nM T68290 CUH90V 23648350 Ki = 133 nM T68290 CCA45G 23648351 Ki = 15 nM T68290 CP10ST 23648352 Ki = 50 nM T68290 CZRA72 23648353 Ki = 208 nM T68290 CPTK56 23648354 Ki = 8 nM T68290 C1YMU6 23648355 Ki = 14 nM T68290 C58JSH 23648356 Ki = 76 nM T68290 C5YS0D 23648357 Ki = 96 nM T68290 CNHA15 23648358 Ki = 15 nM T68290 CQVC57 23648359 Ki = 212 nM T68290 C03ZCQ 23648360 Ki = 12300 nM T68290 CM5QI0 23648361 Ki > 100000 nM T68290 C6YRH9 23648362 Ki > 100000 nM T68290 CP6Q2L 23648363 Ki = 408 nM T68290 C63OZA 23648364 Ki = 70 nM T68290 COU98B 23648365 Ki > 24000 nM T68290 CK43WQ 23648366 Ki = 14 nM T68290 CKQ0P4 23648367 Ki = 18530 nM T68290 CGSN32 23648368 Ki > 100000 nM T68290 C76JKU 23648369 Ki = 15600 nM T68290 C46RQB 23648370 Ki = 226 nM T68290 CPC7Z2 23648371 Ki = 2950 nM T68290 C5FJZ6 23648372 Ki = 143 nM T68290 CL8X1T 23648373 Ki = 100 nM T68290 CL01QA 23648374 Ki = 16 nM T68290 CG9N8B 23648375 Ki = 8 nM T68290 CT98GY 23648376 Ki = 18 nM T68290 CX6JF9 23648377 Ki = 1050 nM T68290 CJ7N9D 23648378 Ki = 80 nM T68290 C0GQ4R 23648379 Ki = 19 nM T68290 CYS7Z2 23648380 Ki = 122 nM T68290 C6H3DY 23648381 Ki = 297 nM T68290 CGV2J8 23648382 Ki = 172 nM T68290 CF0JM1 23648383 Ki = 227 nM T68290 C5LGJ7 23648384 Ki = 217 nM T68290 C39FZB 23648385 Ki = 56 nM T68290 C85STC 23648386 Ki = 39 nM T68290 CWV98T 23648387 Ki = 23 nM T68290 CX59EJ 23648388 Ki = 422 nM T68290 CFNX14 23648389 Ki = 986 nM T68290 CZC34G 23648390 Ki = 1080 nM T68290 C1FJY7 23648391 Ki = 11 nM T68290 C9KW2O 23648392 Ki = 17 nM T68290 CI58TU 23648393 Ki = 213 nM T68290 CB3JX0 23648394 Ki = 18 nM T68290 CYBW67 23648395 Ki = 53 nM T68290 CR1K4V 23648396 Ki = 21 nM T68290 C1B9GH 23648397 Ki = 49 nM T68290 CF72ZM 23648398 Ki = 42 nM T68290 C9X3TS 23648399 Ki = 12 nM T68290 CL8RT9 23648400 Ki = 12 nM T68290 CPEW28 23648401 Ki = 11 nM T68290 CT10OV 23648402 Ki = 11 nM T68290 CEC70K 23648403 Ki = 5 nM T68290 CE2QR4 23648404 Ki = 99 nM T68290 C4F2BY 23648405 Ki = 11400 nM T68290 CX37JK 23648406 Ki = 220 nM T68290 CD8JP5 23648407 Ki = 93 nM T68290 CC7HD5 23648408 Ki = 49 nM T68290 CWGL69 23648409 Ki = 87 nM T68290 CA2DE6 23648410 Ki = 111 nM T68290 C3VT9K 23648411 Ki = 11 nM T68290 CBR76L 23648414 IC50 > 10000 nM T68290 CZ7ME6 23648415 IC50 = 2300 nM T68290 CVU01O 23648416 IC50 = 700 nM T68290 C3M5GX 23648417 IC50 > 10000 nM T68290 CG9NQ8 23648418 IC50 > 10000 nM T68290 C2F1MC 23648419 IC50 > 10000 nM T68290 CCZ4J1 23648420 IC50 = 900 nM T68290 CC2W3A 23648421 IC50 = 969 nM T68290 C8Z5BC 23648422 IC50 = 140 nM T68290 CVD5Y6 23648423 IC50 = 180 nM T68290 CL4Q2D 23648424 IC50 = 52 nM T68290 CF0TY4 23648425 IC50 = 41 nM T68290 CX0V8M 23648426 IC50 = 29 nM T68290 CME4Y9 23648427 IC50 = 130 nM T68290 C4AJB0 23648428 IC50 = 240 nM T68290 C6P3YR 23648430 IC50 = 64 nM T68290 C5AQX8 23648431 IC50 = 35 nM T68290 C0M8FS 23648434 IC50 = 10 nM T68290 CD7R1S 23648435 IC50 = 26 nM T68290 CF9H8N 23648436 IC50 = 15 nM T68290 CZG5U1 23648437 IC50 = 7.9 nM T68290 CF68MH 23648438 IC50 = 10 nM T68290 C2C5YA 23648440 IC50 = 19 nM T68290 C1YTO9 23648449 IC50 = 1373 nM T68290 CN0VA7 24822701 IC50 = 5900 nM T68290 C2GQ6X 24897809 Ki = 0.33 nM T68290 CZ21HD 24898027 Ki = 0.51 nM T68290 CQU38W 24900755 IC50 = 473 nM T68290 C2S8VB 24901099 IC50 = 17 nM T68290 CIN28B 24901100 IC50 = 174 nM T68290 CD2EH0 24901101 IC50 = 298 nM T68290 CS7B3F 24901102 IC50 = 4553 nM T68290 CG9H6V 25008106 IC50 > 1000 nM T68290 CK7BR0 25023784 IC50 = 9 nM T68290 CZH87T 25023785 IC50 = 18 nM T68290 C2PUY3 25023786 IC50 = 9 nM T68290 CFQM73 25023787 IC50 = 11 nM T68290 CTK09I 25023788 IC50 = 5 nM T68290 CDL98C 25023789 IC50 = 17 nM T68290 CCP3G0 25023790 IC50 = 50 nM T68290 CGI0U2 25023791 Ki = 4 nM T68290 CY4TR2 25024777 IC50 = 790 nM T68290 CM56PL 25024778 IC50 = 610 nM T68290 CB8WL6 25024779 IC50 = 480 nM T68290 CB0R9F 25024979 IC50 = 1500 nM T68290 CO5U3T 25026563 IC50 = 580 nM T68290 CO72TX 25027584 IC50 = 2 nM T68290 C8CIY2 25030810 IC50 = 6 nM T68290 CMS0L3 25052748 IC50 = 13 nM T68290 C7J3MN 25053851 IC50 > 1000 nM T68290 C6AVL9 25053852 IC50 > 1000 nM T68290 C19GML 25071954 IC50 < 1 nM T68290 C5D3HC 25102859 IC50 = 130 nM T68290 C5BR1Q 25102865 IC50 = 420 nM T68290 C0JAF3 25102978 IC50 = 80 nM T68290 C5C6XF 25102980 IC50 = 460 nM T68290 CUX5I1 25102981 IC50 = 360 nM T68290 CIEV95 25102982 IC50 = 530 nM T68290 CR2TI8 25103094 IC50 = 1280 nM T68290 C7D9OJ 25103218 IC50 = 380 nM T68290 CNJI51 25103579 IC50 = 2010 nM T68290 CM1VK0 25103581 IC50 = 560 nM T68290 C7QPU8 25103705 IC50 = 470 nM T68290 C53VOM 25103706 IC50 = 810 nM T68290 C3WGF1 25103831 IC50 = 380 nM T68290 C5QS8O 25103833 IC50 = 30 nM T68290 C49SCW 25104073 IC50 = 100 nM T68290 C2YRL1 25104074 IC50 = 340 nM T68290 C0B8WC 25104315 IC50 = 350 nM T68290 CC62YP 25104316 IC50 = 40 nM T68290 C8Q1VW 25104319 IC50 = 1150 nM T68290 CYAN35 25104321 IC50 = 210 nM T68290 CZ3NT9 25104322 IC50 = 60 nM T68290 CUR2G8 25104435 IC50 = 20 nM T68290 CO2CD5 25104437 IC50 = 370 nM T68290 C42KMB 25104547 IC50 = 160 nM T68290 C9YO1X 25104549 IC50 = 200 nM T68290 CZU49J 25104658 IC50 = 270 nM T68290 CPGT89 25104661 IC50 = 800 nM T68290 CGFQ91 25104663 IC50 = 130 nM T68290 C8H1PT 25104665 IC50 = 390 nM T68290 CF54QZ 25129041 IC50 = 1584.89 nM T68290 CDO26T 25129042 IC50 = 630.96 nM T68290 C57LJM 25129043 IC50 = 1370 nM T68290 C3AT6W 25130088 IC50 = 1250 nM T68290 C1FWI6 25133836 IC50 = 2150 nM T68290 CYV1J6 25133837 IC50 > 7430 nM T68290 CBZK08 25133838 IC50 = 3162.28 nM T68290 CP8U3Q 25142042 IC50 > 4000 nM T68290 CC92AI 25142043 IC50 > 4000 nM T68290 C8IFW0 25142172 IC50 > 4000 nM T68290 CD2A6W 25142173 IC50 > 4000 nM T68290 C53OMA 25142175 IC50 > 4000 nM T68290 C7CFR2 25142176 IC50 > 4000 nM T68290 C78RJG 25142177 IC50 > 4000 nM T68290 CS6R4T 25142308 IC50 > 4000 nM T68290 CM2PI4 25142309 IC50 > 4000 nM T68290 CM6FL3 25142310 IC50 > 4000 nM T68290 CWV4F5 25142312 IC50 > 4000 nM T68290 CH52AJ 25142313 IC50 > 4000 nM T68290 COG9V7 25142440 IC50 > 4000 nM T68290 CYL56K 25142444 IC50 > 4000 nM T68290 C3IT4O 25142445 IC50 > 4000 nM T68290 CK7D0V 25142571 IC50 > 4000 nM T68290 CW9KR5 25142573 IC50 > 4000 nM T68290 CZ0G2I 25142574 IC50 > 4000 nM T68290 CNH31I 25142699 IC50 > 4000 nM T68290 CQ9PD6 25142700 IC50 > 4000 nM T68290 CV08DB 25142970 IC50 > 4000 nM T68290 C3C8YJ 25174148 IC50 = 1000 nM T68290 C5M1BT 25195691 IC50 = 3981.07 nM T68290 CTLO73 25204268 IC50 = 28 nM T68290 C42ZMF 25204335 IC50 = 9.5 nM T68290 CC7TV3 25204336 IC50 = 63 nM T68290 CFX41G 25204403 IC50 = 20 nM T68290 CU59SO 25242431 Ki = 0.7 nM T68290 C23JPC 25242432 Ki = 1 nM T68290 C6Y0ME 25242511 IC50 = 0.6 nM T68290 CW9JM2 25256832 IC50 = 560 nM T68290 C3GC7P 25256833 IC50 = 890 nM T68290 CXEZ30 25266292 IC50 = 2 nM T68290 CZS24P 42633520 IC50 = 408 nM T68290 CI78XT 42633521 IC50 = 322 nM T68290 CZ6B1F 42635119 IC50 = 169 nM T68290 CZM36T 42641892 IC50 > 10000 nM T68290 CRYH80 42642459 IC50 > 10000 nM T68290 C3DC4M 42647278 Ki = 0.56 nM T68290 C25ELB 44143088 IC50 = 15.85 nM T68290 CL0M7R 44143089 IC50 = 26915.35 nM T68290 C9QDC0 44143091 IC50 = 104.71 nM T68290 CLPN48 44192275 IC50 = 420 nM T68290 C1YS3D 44192358 IC50 = 350 nM T68290 CH9RV1 44192359 IC50 = 510 nM T68290 CE7F0J 44192360 IC50 = 90 nM T68290 C6OTZ8 44192361 IC50 = 190 nM T68290 C1DQ0B 44192445 IC50 = 80 nM T68290 C03TJW 44192539 IC50 = 820 nM T68290 C6KUC8 44192634 IC50 = 50 nM T68290 C8C9KL 44224000 IC50 = 220 nM T68290 CJA68L 44224113 IC50 = 125.89 nM T68290 C2V5ZT 44224114 IC50 = 2511.89 nM T68290 C0U9VJ 44224115 IC50 = 1995.26 nM T68290 C0MZ9D 44224116 IC50 = 2511.89 nM T68290 CEJ82A 44224117 IC50 = 630.96 nM T68290 C0KL7D 44224118 IC50 = 398.11 nM T68290 CE9S0M 44224119 IC50 = 1584.89 nM T68290 CV1W0Z 44224120 IC50 = 199.53 nM T68290 C5LDK7 44224121 IC50 = 1258.93 nM T68290 C8UF5Q 44224122 IC50 = 1995.26 nM T68290 C9YHC5 44224123 IC50 = 316.23 nM T68290 CA26RI 44224124 IC50 = 3162.28 nM T68290 CU0PI2 44224125 IC50 > 10000 nM T68290 CRL79W 44224126 IC50 = 3162.28 nM T68290 C3T0QO 44224127 IC50 = 1000 nM T68290 C81EVM 44224128 IC50 = 1258.93 nM T68290 C7IY8P 44224129 IC50 = 794.33 nM T68290 CYG02V 44224130 IC50 = 794.33 nM T68290 CJS1B9 44224131 IC50 = 199.53 nM T68290 CN5O8S 44224132 IC50 = 794.33 nM T68290 C2Q3RP 44224133 IC50 = 794.33 nM T68290 CZX62T 44224134 IC50 = 794.33 nM T68290 CP3YA9 44224135 IC50 = 1000 nM T68290 CSZH31 44224136 IC50 = 794.33 nM T68290 CI3LU0 44263386 IC50 = 7900 nM T68290 C6A1BZ 44263387 IC50 = 11000 nM T68290 CV54MF 44263388 IC50 = 8300 nM T68290 CUG31X 44263389 IC50 = 6700 nM T68290 C3I4CN 44263390 IC50 = 1500 nM T68290 CH3E1I 44263392 IC50 = 720 nM T68290 CWR61C 44263393 IC50 = 1100 nM T68290 COH24Y 44263394 IC50 = 870 nM T68290 CR6IF4 44263395 IC50 = 550 nM T68290 CD2P3H 44263396 IC50 = 700 nM T68290 CGNF32 44263397 IC50 = 1500 nM T68290 CZ56BP 44263398 IC50 = 200 nM T68290 C1V4BN 44263399 IC50 = 280 nM T68290 C3CRK6 44263400 IC50 = 280 nM T68290 CT0OR2 44263401 IC50 = 430 nM T68290 C2VQS7 44263402 IC50 = 510 nM T68290 CT3IY4 44263403 IC50 = 320 nM T68290 C45FSQ 44263404 IC50 = 140 nM T68290 C5FDI4 44263405 IC50 = 330 nM T68290 C8C7AG 44263406 IC50 = 310 nM T68290 C7LS9Z 44263407 IC50 = 280 nM T68290 CR38EU 44279051 Ki = 26 nM T68290 CD84XF 44279475 IC50 = 2500 nM T68290 CFJ2Z1 44279771 IC50 = 330 nM T68290 C3IBQ0 44279792 IC50 > 2500 nM T68290 CQ57HR 44279823 IC50 = 355 nM T68290 C5YF0J 44279873 IC50 > 5000 nM T68290 C6ZXK0 44280152 IC50 = 20 nM T68290 CVZ54E 44280172 IC50 = 41 nM T68290 C2ZHC1 44295739 IC50 > 10000 nM T68290 CNL8Y4 44302956 IC50 = 470 nM T68290 CAM2S5 44302974 IC50 = 5800 nM T68290 CBYD40 44302975 IC50 = 480 nM T68290 CNA24Z 44303031 IC50 = 1200 nM T68290 C56IEO 44303058 IC50 = 1200 nM T68290 CL4VM1 44303061 IC50 = 1100 nM T68290 CS0P5A 44303274 IC50 > 10000 nM T68290 CXU16T 44303285 IC50 = 4400 nM T68290 CEIH70 44303290 IC50 = 9500 nM T68290 CN21AS 44303309 IC50 = 5700 nM T68290 C24EDH 44303315 IC50 = 4600 nM T68290 CDX5M7 44303318 IC50 = 4500 nM T68290 CRK48P 44303319 IC50 = 7500 nM T68290 CKB9O1 44303324 IC50 = 4900 nM T68290 C0FEJ1 44303335 IC50 = 580 nM T68290 CT49MJ 44303338 IC50 = 320 nM T68290 CMF6W2 44303344 IC50 = 660 nM T68290 CD1HJ5 44303345 IC50 = 480 nM T68290 CL26OE 44303389 IC50 = 160 nM T68290 CN9QY5 44303414 IC50 = 3400 nM T68290 CG3OM8 44304535 Ki = 33000 nM T68290 C0FKB3 44304563 Ki = 28000 nM T68290 CC04TQ 44304591 Ki > 150000 nM T68290 C76OIY 44304610 Ki = 130 nM T68290 CK8JW5 44304611 Ki = 20000 nM T68290 CZ87NW 44304634 Ki = 11000 nM T68290 COR96D 44304861 Ki = 53000 nM T68290 CKB02C 44329582 Ki = 451 nM T68290 CTN34G 44329585 Ki = 460 nM T68290 CR1J6F 44329593 Ki = 811 nM T68290 C3EHF1 44329596 Ki = 88 nM T68290 C97WPV 44329608 Ki = 110 nM T68290 CY5KH4 44329643 Ki = 4500 nM T68290 C7MWQ8 44342499 IC50 = 8 nM T68290 CQ61OB 44342501 IC50 = 2500 nM T68290 CIBF96 44342511 IC50 = 4.6 nM T68290 CVK4H3 44342519 IC50 = 3 nM T68290 CN7BH9 44342744 IC50 > 2500 nM T68290 CP2OM5 44342745 IC50 = 0.7 nM T68290 CMQ6Y0 44342776 IC50 = 260 nM T68290 C6PLY0 44342983 IC50 = 70 nM T68290 C8HP5M 44347822 IC50 = 2364 nM T68290 CK0B9C 44347827 IC50 > 10000 nM T68290 CO82ZV 44347993 IC50 > 10000 nM T68290 CLCP51 44348116 IC50 = 3368 nM T68290 CFBI42 44348134 IC50 = 1748 nM T68290 CYEI89 44348185 IC50 = 521 nM T68290 CNZ2I9 44353889 IC50 = 1000 nM T68290 C9EOS5 44353924 IC50 > 1000 nM T68290 CG1JP8 44353951 IC50 = 1000 nM T68290 CX1IL0 44353974 IC50 = 1200 nM T68290 CQ1F6V 44353976 IC50 = 780 nM T68290 CJA79K 44353977 IC50 > 1000 nM T68290 C3GV4U 44353978 IC50 = 1700 nM T68290 C67ZFU 44353986 IC50 = 3900 nM T68290 CT7JK8 44354015 IC50 = 710 nM T68290 C49VSE 44354016 IC50 = 2600 nM T68290 C4D9RS 44367595 IC50 = 387 nM T68290 CV49WI 44390016 IC50 = 190 nM T68290 CH6J2L 44390026 IC50 = 350 nM T68290 C2Q8DK 44390039 IC50 = 200 nM T68290 CSDE03 44390040 IC50 = 180 nM T68290 CIG5R6 44393795 IC50 = 897 nM T68290 CTRP74 44394287 IC50 = 270 nM T68290 CP7X6J 44394353 IC50 = 20 nM T68290 C79NFU 44394458 IC50 = 430 nM T68290 CKWV17 44396536 IC50 = 5 nM T68290 C2J6MW 44397423 IC50 = 810 nM T68290 CRSF50 44397609 IC50 = 540 nM T68290 CHWX97 44397693 IC50 = 2700 nM T68290 CZC50Y 44398247 IC50 > 10000 nM T68290 CQPM06 44398248 IC50 > 10000 nM T68290 CYJ8Z4 44398353 IC50 = 340 nM T68290 CD18YP 44402055 IC50 = 79 nM T68290 CU8TB9 44402056 IC50 = 16 nM T68290 CD4TP7 44402158 IC50 = 280 nM T68290 CO6BG2 44402160 IC50 = 30 nM T68290 C0AJC4 44402175 IC50 = 290 nM T68290 CX9O2Q 44402263 IC50 = 63 nM T68290 C89MOT 44402291 IC50 = 19 nM T68290 CFL9B8 44402952 IC50 = 902 nM T68290 CRZT97 44403028 IC50 > 10000 nM T68290 CW2L5D 44404573 Ki = 3707 nM T68290 C39PTS 44404574 Ki = 6769 nM T68290 CY5NW9 44405210 Ki = 10000 nM T68290 CP8L2A 44405213 Ki = 4500 nM T68290 CA59MJ 44405279 Ki = 400 nM T68290 C5GS4Y 44405280 Ki = 4200 nM T68290 CDP93F 44405305 Ki = 42000 nM T68290 C9IEW7 44409018 Ki = 16 nM T68290 CFD89M 44410036 IC50 = 322 nM T68290 C5RTQ8 44410054 IC50 = 1775 nM T68290 CS1NY3 44410075 IC50 = 75 nM T68290 CTC4X1 44410206 IC50 = 1700 nM T68290 CR04PA 44410374 IC50 = 900 nM T68290 C21GXN 44410779 Ki = 46 nM T68290 CY4H2I 44411981 Ki = 300 nM T68290 CNU4T9 44412155 Ki < 0.25 nM T68290 CYF1B9 44412339 Ki = 19000 nM T68290 C1J6OW 44412340 Ki = 130000 nM T68290 CU49OM 44412341 Ki = 12000 nM T68290 CDK32G 44412349 Ki = 800 nM T68290 CL82XD 44412354 Ki = 2600 nM T68290 C23ZVR 44412355 Ki = 2000 nM T68290 CV26BC 44412365 Ki = 380 nM T68290 CX93NW 44412366 Ki = 240 nM T68290 CZN9T0 44412387 Ki = 320 nM T68290 CY90QW 44412402 Ki = 760 nM T68290 C1HW8F 44412424 Ki = 140 nM T68290 CYDJ14 44412436 Ki = 700 nM T68290 CV49GB 44412437 Ki = 9200 nM T68290 CZ5VW2 44412440 Ki = 960 nM T68290 CZR1O3 44412502 Ki = 28000 nM T68290 CA23SL 44414977 Ki = 9500 nM T68290 C0XB2M 44414978 Ki = 5600 nM T68290 CAG5F3 44414992 Ki = 7400 nM T68290 C8JL9C 44415006 Ki = 3600 nM T68290 CS6X7V 44426055 IC50 = 696 nM T68290 C8IB2W 44426056 IC50 > 100000 nM T68290 CBI1A2 44430130 IC50 = 171 nM T68290 CP9EX2 44430136 IC50 = 37 nM T68290 CD1QV3 44430138 IC50 = 62 nM T68290 CT62BZ 44430168 IC50 = 135 nM T68290 CRP21Y 44430178 IC50 = 251 nM T68290 C5T0CN 44430196 IC50 = 207 nM T68290 C8OP1X 44430245 IC50 = 141 nM T68290 C01JVR 44430250 IC50 = 155 nM T68290 C4VD7O 44430252 IC50 = 66 nM T68290 CC4WZ2 44430254 IC50 = 39 nM T68290 CN5RW8 44430256 IC50 = 22 nM T68290 C5J4AD 44430257 IC50 = 75 nM T68290 C5G6AM 44430258 IC50 = 23 nM T68290 CCI24L 44430259 IC50 = 41 nM T68290 CF5B8S 44430260 IC50 = 23 nM T68290 CDYE46 44430261 IC50 = 29 nM T68290 C1KJ6M 44430262 IC50 = 22.32 nM T68290 C81PIB 44430263 IC50 = 47 nM T68290 C92NCW 44430264 IC50 = 14 nM T68290 CACS87 44430265 IC50 = 1.9 nM T68290 C8FE5D 44430266 IC50 = 3136 nM T68290 CM83FJ 44430267 IC50 = 63 nM T68290 CK4FY6 44430268 IC50 = 42 nM T68290 C86FHS 44433594 IC50 = 290 nM T68290 C6V1EB 44433598 IC50 = 1800 nM T68290 CEKY65 44433599 IC50 = 370 nM T68290 CVD7L4 44442257 IC50 = 2237 nM T68290 CFN67O 44444198 IC50 = 390 nM T68290 C24AIO 44444199 IC50 = 490 nM T68290 CCM4R1 44444200 IC50 > 1000 nM T68290 CR3DP0 44444201 IC50 = 980 nM T68290 CN5OJ8 44444202 IC50 = 730 nM T68290 CRJ07X 44444203 IC50 = 100 nM T68290 CSUC26 44444204 IC50 = 930 nM T68290 C3J4DH 44444205 IC50 = 460 nM T68290 C5T1NC 44444208 IC50 = 820 nM T68290 CGCU82 44444211 IC50 > 1000 nM T68290 CGB81X 44444216 IC50 > 1000 nM T68290 C9VB5M 44444217 IC50 = 320 nM T68290 C8FN2V 44444218 IC50 > 1000 nM T68290 C1L9BM 44444221 IC50 > 1000 nM T68290 CZ25FP 44444222 IC50 = 160 nM T68290 CTW39N 44444223 IC50 = 220 nM T68290 C6J8LS 44444224 IC50 = 440 nM T68290 CW2L4V 44444225 IC50 > 1000 nM T68290 CA9JR0 44444228 IC50 > 1000 nM T68290 CTQ81M 44444229 IC50 > 1000 nM T68290 CWE50F 44444230 IC50 > 1000 nM T68290 CT8QV6 44444231 IC50 > 1000 nM T68290 CISQ24 44444232 IC50 > 1000 nM T68290 C8CQS6 44444233 IC50 > 1000 nM T68290 CP79CA 44444234 IC50 > 1000 nM T68290 CXO56L 44447657 IC50 = 2834 nM T68290 CB6H5U 44447658 IC50 = 2489 nM T68290 C1U6JA 44447659 IC50 = 266 nM T68290 CV3T1A 44447660 IC50 > 10000 nM T68290 CF7AV1 44447661 IC50 = 56 nM T68290 C7HRP2 44447662 IC50 = 170 nM T68290 C0CZ7P 44447663 IC50 = 17 nM T68290 CAF54M 44447664 IC50 = 15 nM T68290 CC4J7S 44447665 IC50 = 89 nM T68290 CL6WZ1 44450271 IC50 = 760 nM T68290 C3B2TR 44450349 IC50 > 1000 nM T68290 C38JBH 44450361 IC50 > 1000 nM T68290 CZG3F8 44452745 Ki < 100 nM T68290 CN70AJ 44452769 Ki < 100 nM T68290 CC0AG3 44452909 Ki = 40 nM T68290 CB8IX2 44452912 Ki = 30 nM T68290 CVCJ36 44452938 Ki < 0.25 nM T68290 C4ZBF6 44452963 Ki = 2000 nM T68290 CWCK10 44452964 Ki = 380 nM T68290 CF9PC3 44452965 Ki = 26000 nM T68290 C49IHD 44453066 Ki < 10 nM T68290 C8Z4WO 44459967 IC50 = 6456.54 nM T68290 C86ORE 44459987 IC50 = 5623.41 nM T68290 C9TFJ8 44464926 IC50 = 1995.26 nM T68290 CYO0T1 44465454 IC50 = 316.23 nM T68290 CE83YL 44465721 IC50 = 125.89 nM T68290 CV1IL5 44565796 IC50 = 910 nM T68290 CI6H7R 44568190 IC50 = 16 nM T68290 CVX81T 44568191 IC50 = 6 nM T68290 CJRQ74 44568192 IC50 = 7 nM T68290 C6ZHA4 44568193 IC50 = 2 nM T68290 C2X3HJ 44568223 IC50 = 8 nM T68290 CV54EU 44568306 IC50 = 12 nM T68290 CDZ03Q 44568307 IC50 = 15 nM T68290 C6FV7W 44568638 IC50 = 320 nM T68290 C6U3RB 44568639 IC50 = 110 nM T68290 COJ16S 44568640 IC50 = 21 nM T68290 CVP4Y6 44568641 IC50 = 150 nM T68290 CZW5K2 44568669 IC50 = 7 nM T68290 CW89JM 44568670 IC50 = 33 nM T68290 C2D9TS 44568671 IC50 = 99 nM T68290 CU4PO0 44568672 IC50 = 64 nM T68290 CCJ68F 44568673 IC50 = 19 nM T68290 CCIP49 44568714 IC50 = 190 nM T68290 C3HYW8 44568715 IC50 > 1000 nM T68290 CLXN21 44568716 IC50 = 110 nM T68290 C40KFC 44568717 IC50 = 440 nM T68290 CA86UV 44568718 IC50 = 140 nM T68290 CU82VX 44568766 IC50 = 24 nM T68290 CZF5G0 44568767 IC50 = 52 nM T68290 CVR02S 44568768 IC50 = 10 nM T68290 C1P3LN 44568769 IC50 = 11 nM T68290 CG74ZL 44568770 IC50 = 6 nM T68290 COHB20 44570671 Ki = 2.4 nM T68290 C35ZYP 44570672 Ki = 180 nM T68290 C3BHM4 44570673 Ki = 5.3 nM T68290 C0OSY2 44570674 Ki = 0.8 nM T68290 CF41YI 44570719 Ki = 31 nM T68290 CY9ZT4 44570833 Ki = 26 nM T68290 CB3S2D 44570834 Ki = 330 nM T68290 C8K6PB 44570835 Ki = 4.9 nM T68290 CWH9Q0 44570836 Ki = 30 nM T68290 CA10KC 44570876 Ki = 5.6 nM T68290 CAUD26 44570877 Ki = 16 nM T68290 C1XCP6 44570878 Ki = 57 nM T68290 CN1GT2 44570879 Ki = 4 nM T68290 CV0KJ4 44570915 Ki = 12 nM T68290 C14JNH 44570916 Ki = 56 nM T68290 C1DA8K 44570917 Ki = 63 nM T68290 C9CMZ2 44570957 Ki = 2 nM T68290 C37LRT 44570958 Ki = 3.4 nM T68290 C31BXW 44570959 Ki = 3.8 nM T68290 C5G2KT 44570997 Ki = 3.9 nM T68290 CZ1ET3 44570998 Ki = 1.3 nM T68290 CSYI14 44570999 Ki = 3.3 nM T68290 CK5ZM6 44571085 Ki = 1.1 nM T68290 CNP2G3 44571086 Ki = 0.6 nM T68290 CX2B3F 44571130 Ki = 0.8 nM T68290 CFTE86 44571131 Ki = 2.7 nM T68290 C4DV1E 44571132 Ki = 2.1 nM T68290 C05LYD 44571173 Ki = 2.3 nM T68290 CC5A6D 44571174 Ki = 0.9 nM T68290 CHB7Y3 44571175 Ki = 5.9 nM T68290 C6XF8B 44571212 Ki = 2.3 nM T68290 CG5ZO3 44571213 Ki = 4.5 nM T68290 C67UMF 44571214 Ki = 13 nM T68290 CD6X2Y 44571254 Ki = 5.7 nM T68290 CQ0W5J 44571255 Ki = 8.6 nM T68290 CGM30J 44571297 Ki = 31 nM T68290 CU0D3P 44571298 Ki = 2.6 nM T68290 CUG72S 44571323 Ki = 12 nM T68290 C2NT4H 44571324 Ki = 110 nM T68290 CC12QS 44571325 Ki = 140 nM T68290 CI39YN 44571326 Ki = 190 nM T68290 C1L3KX 44571358 Ki = 1.9 nM T68290 C0NFJ8 44571359 Ki = 3.4 nM T68290 CE2PQ4 44571360 Ki = 8.3 nM T68290 C5S6FJ 44571361 Ki = 2.9 nM T68290 C9E6QP 44579079 IC50 = 31 nM T68290 C7CKG9 44579080 IC50 = 12 nM T68290 CFN0Z1 44579081 IC50 > 1000 nM T68290 CH5B0N 44579120 IC50 = 4 nM T68290 CN42GY 44579121 IC50 = 3 nM T68290 CDUJ10 44579122 IC50 = 26 nM T68290 CQJ0L6 44579123 IC50 = 3 nM T68290 CO13BP 44579170 IC50 = 3 nM T68290 CP0X4D 44579171 IC50 = 5 nM T68290 CS60PG 44579172 IC50 = 5 nM T68290 CY2E6M 44579173 IC50 = 10 nM T68290 CA0OT2 44587365 IC50 < 1 nM T68290 CM35BH 44587366 IC50 < 1 nM T68290 C2AVQ0 44587440 IC50 = 22 nM T68290 CO7TR5 44587827 IC50 = 22 nM T68290 CL18MT 44587828 IC50 = 32 nM T68290 C3A4JO 44587829 IC50 = 14 nM T68290 C9HES8 44587858 IC50 = 22 nM T68290 CA4DK2 44587859 IC50 = 93 nM T68290 C76PSY 44587860 IC50 = 15 nM T68290 C6NU0J 44587861 IC50 = 24 nM T68290 C8C1OM 44587862 IC50 = 3 nM T68290 CERA06 44587897 IC50 = 23 nM T68290 CI87JG 44587898 IC50 = 4 nM T68290 C2OQE5 44587899 IC50 = 21 nM T68290 CNM2G4 44587937 IC50 = 6 nM T68290 C65NLR 44587938 IC50 = 7 nM T68290 C81ZSB 44587939 IC50 = 1 nM T68290 CBW29L 45139235 IC50 = 80 nM T68290 C8F1UP 45482747 IC50 = 40 nM T68290 CJ9W7Q 45482764 IC50 = 7400 nM T68290 C58YWJ 45482785 IC50 = 140 nM T68290 C94QTO 45482786 IC50 = 150 nM T68290 CSA23B 45482804 IC50 = 380 nM T68290 CG8F6W 45482816 IC50 = 80 nM T68290 CGJ13N 45482817 IC50 = 20 nM T68290 CD80CY 45482818 IC50 = 110 nM T68290 CCNP30 45482844 IC50 = 490 nM T68290 C61TSM 45482845 IC50 = 160 nM T68290 C5RWY6 45482846 IC50 = 350 nM T68290 CVC03H 45482858 IC50 = 1300 nM T68290 CNJF96 45482859 IC50 = 600 nM T68290 CU37FT 45482860 IC50 = 100 nM T68290 CSI14H 45482861 IC50 = 100 nM T68290 C6JH1V 45482862 IC50 = 120 nM T68290 CBA0G4 45482863 IC50 = 10 nM T68290 CAM56H 45482864 IC50 = 30 nM T68290 CW07MH 45482865 IC50 = 10 nM T68290 CQ53LK 45482866 IC50 = 720 nM T68290 C3DRB6 45496892 IC50 > 200000 nM T68290 C6JP8Z 46174174 IC50 = 40 nM T68290 C71ABD 46174175 IC50 = 430 nM T68290 C4YAJ7 46228924 IC50 = 78000 nM T68290 C5QE7P 46238539 IC50 = 58 nM T68290 CJ64BK 46830170 IC50 = 110 nM T68290 CU2JY5 46830171 IC50 = 55 nM T68290 CH7YV9 46830172 IC50 = 160 nM T68290 CB4TH2 46830192 IC50 = 10 nM T68290 CD74CL 46830193 IC50 = 90 nM T68290 CAX1J2 46830194 IC50 = 40 nM T68290 C9MJ3F 46830240 IC50 = 3920 nM T68290 CH2TL9 46830241 IC50 = 190 nM T68290 CYO3F7 46830256 IC50 = 380 nM T68290 CWJP64 46830257 IC50 = 10 nM T68290 C7KB8E 46830803 IC50 = 8.8 nM T68290 C05ZYX 46834545 IC50 = 6.6 nM T68290 CC2N0F 46842579 IC50 = 39 nM T68290 CV6SW4 46842581 IC50 = 3.3 nM T68290 CM2D1G 46842582 IC50 = 8.3 nM T68290 CIU1R5 46842626 IC50 = 18.6 nM T68290 C37OSC 46842709 IC50 = 14.1 nM T68290 C6HD4M 46865101 IC50 > 10000 nM T68290 CC7DG3 46866398 IC50 = 20 nM T68290 CWL1T4 46871744 IC50 = 5.8 nM T68290 C38HWY 46878211 Ki > 3000 nM T68290 CZ43KH 46878212 Ki > 3000 nM T68290 CGT1Z2 46881448 IC50 = 191 nM T68290 CH9ON3 46881449 IC50 = 155 nM T68290 CF15KQ 46881450 IC50 = 93 nM T68290 CJ0XH5 46881452 IC50 = 191 nM T68290 C6O2JN 46881453 IC50 > 10000 nM T68290 CN58BG 46882092 IC50 = 41 nM T68290 CG9X3C 46882094 IC50 > 10000 nM T68290 CZ5KP8 46882095 IC50 = 1259 nM T68290 CPQZ83 46882096 IC50 = 28 nM T68290 CHX21M 46882097 IC50 = 1047 nM T68290 CDYJ19 46884237 IC50 = 1650 nM T68290 C1KQ0O 46884238 IC50 = 1470 nM T68290 CE2NW3 46884272 IC50 = 3600 nM T68290 C6B0FX 46884273 IC50 = 600 nM T68290 CDF4J8 46884274 IC50 = 740 nM T68290 CFD4A9 46884275 IC50 = 220 nM T68290 CQ86BX 46884276 IC50 = 200 nM T68290 C1PF4X 46884277 IC50 = 960 nM T68290 CL72RZ 46884333 IC50 = 335 nM T68290 C8K2JA 46884334 IC50 = 335 nM T68290 C16MXY 46884335 IC50 = 325 nM T68290 C5IUJ6 46884336 IC50 = 595 nM T68290 C7QOU2 46884337 IC50 = 1150 nM T68290 C2WH3Q 46884338 IC50 = 220 nM T68290 C5J2BG 46884339 IC50 = 81 nM T68290 CRQ5Y0 46884340 IC50 = 710 nM T68290 CFMC24 46884341 IC50 = 1130 nM T68290 CI6XP9 46884342 IC50 = 420 nM T68290 CHA3I0 46884343 IC50 = 712 nM T68290 C7FB1I 46884344 IC50 = 1035 nM T68290 CTE1O7 46884345 IC50 = 565 nM T68290 C5IX6R 46884346 IC50 = 149 nM T68290 CW3I1H 46884347 IC50 = 395 nM T68290 CYKV72 46884348 IC50 = 58 nM T68290 CH9T0F 46884378 IC50 = 9600 nM T68290 C5HXY2 46884379 IC50 = 9000 nM T68290 CPQH87 46884380 IC50 = 350 nM T68290 CS14ZU 46884381 IC50 = 300 nM T68290 C20KBI 46884382 IC50 = 235 nM T68290 C6HRV5 46884383 IC50 = 1190 nM T68290 C39YIQ 46884384 IC50 = 355 nM T68290 CSO23Q 46884385 IC50 = 205 nM T68290 CB1FS9 46884386 IC50 = 385 nM T68290 CK09YO 46884387 IC50 = 690 nM T68290 CHK48E 46884388 IC50 = 235 nM T68290 C6YGQ0 46884389 IC50 = 245 nM T68290 CA6SF3 46884390 IC50 = 470 nM T68290 C5LN0Z 46884391 IC50 = 310 nM T68290 CJDU43 46884392 IC50 = 810 nM T68290 CVXU89 46884393 IC50 = 70 nM T68290 C2OS0G 46884489 IC50 = 60 nM T68290 CZ0HW4 46884490 IC50 = 250 nM T68290 C7GYF6 46884491 IC50 = 110 nM T68290 C5DTR1 46884492 IC50 = 30 nM T68290 CA5XO1 46884493 IC50 = 1540 nM T68290 CC41BM 46884494 IC50 = 10000 nM T68290 CBL2V8 46884495 IC50 = 470 nM T68290 CZ0X9B 46884496 IC50 = 7 nM T68290 C3R7OD 46884497 IC50 = 20 nM T68290 CPOV20 46884498 IC50 = 40 nM T68290 C6NZF1 46884499 IC50 = 10 nM T68290 C75QIM 46884500 IC50 = 3130 nM T68290 CDGW63 46884501 IC50 = 110 nM T68290 CV36IO 46884502 IC50 = 520 nM T68290 C5CYU0 46884503 IC50 = 520 nM T68290 CSZ75G 46884504 IC50 = 110 nM T68290 C5I1NO 46884505 IC50 = 60 nM T68290 C2YJV1 46884506 IC50 = 190 nM T68290 CVQK72 46884507 IC50 = 900 nM T68290 C7HPI9 46884508 IC50 = 10 nM T68290 CS98EA 46891067 IC50 = 3.1 nM T68290 C2DLA8 46891068 IC50 = 8 nM T68290 C0IW4D 46891069 IC50 = 2 nM T68290 CWCD72 46891070 IC50 = 3.6 nM T68290 CSU14E 46891071 IC50 = 3.8 nM T68290 C52GQT 46891072 IC50 = 7.2 nM T68290 CIQ02Z 46891073 IC50 = 10.3 nM T68290 CZHQ53 46891121 IC50 = 3.4 nM T68290 CNS43V 46891122 IC50 = 4.3 nM T68290 C7A0YQ 46891123 IC50 = 49.2 nM T68290 CSLP13 46891124 IC50 = 15.7 nM T68290 CDH52G 46891125 IC50 = 2.1 nM T68290 CG1N7D 46891126 IC50 > 100 nM T68290 CT2YK4 46891127 IC50 > 100 nM T68290 CK97YW 46891128 IC50 = 5.6 nM T68290 CE95GU 46891129 IC50 = 6.2 nM T68290 CMSC16 46891130 IC50 = 5.9 nM T68290 CE5S7P 46891131 IC50 = 11.5 nM T68290 CFA06V 46891132 IC50 = 23.8 nM T68290 C7C3ND 46891133 IC50 = 6.2 nM T68290 C7F2PT 46891134 IC50 = 2.3 nM T68290 CO0MS2 46891135 IC50 = 6.1 nM T68290 CQIH87 46891136 IC50 = 42.3 nM T68290 C3E5ZS 46891137 IC50 = 5.7 nM T68290 CWO8D9 46891138 IC50 = 7.1 nM T68290 CQ2D0R 46891139 IC50 = 22.8 nM T68290 CUV3G7 46891177 IC50 = 4.4 nM T68290 CJH26Z 46891178 IC50 = 1.9 nM T68290 CUI91D 46905615 IC50 = 1600 nM T68290 C50BXV 46911628 IC50 = 31 nM T68290 CYG6M1 46911633 IC50 = 3.9 nM T68290 CTW1Q2 46911634 IC50 = 7.2 nM T68290 C07GBO 46911635 IC50 = 6.9 nM T68290 C4SWM6 46911715 IC50 = 60 nM T68290 CFWU08 46946224 IC50 = 2 nM T68290 CVT40A 46947220 IC50 = 1 nM T68290 CAFW31 49783666 IC50 > 10000 nM T68290 CI7P2B 49797571 IC50 = 33400 nM T68290 CI59MV 49797572 IC50 > 50000 nM T68290 C96CKU 49797573 IC50 = 5900 nM T68290 CIE60C 49797973 IC50 = 14000 nM T68290 CJ9V8G 49797974 IC50 = 1600 nM T68290 CBE7Q8 49797975 IC50 = 2300 nM T68290 CH91CN 49797976 IC50 = 1500 nM T68290 CW6KB3 49797977 IC50 = 320 nM T68290 CX2BD8 49797978 IC50 = 110 nM T68290 C4NB3R 49834903 IC50 = 0.8 nM T68290 CQ3W9J 49834904 IC50 = 1 nM T68290 CX1WU8 49834905 IC50 = 11 nM T68290 CA96LF 49834906 IC50 = 7 nM T68290 CB9MS2 49834907 IC50 = 0.4 nM T68290 C74RAF 49834908 IC50 = 1 nM T68290 CN8E2A 49834971 IC50 = 0.5 nM T68290 COG9T6 49834972 IC50 = 4 nM T68290 CGPM91 49834975 IC50 = 2 nM T68290 CJ73DH 49835032 IC50 = 10 nM T68290 C8XR4Q 49835033 IC50 = 2 nM T68290 CXE51M 49835035 IC50 = 6 nM T68290 CKRG17 49835144 IC50 = 3 nM T68290 C9NO4U 49835145 IC50 = 4 nM T68290 CS23QM 49835147 IC50 = 0.9 nM T68290 CCO0S5 49835202 IC50 = 230 nM T68290 CP4S5A 49835673 IC50 = 0.7 nM T68290 CS3HC6 49835674 IC50 = 0.7 nM T68290 CSTC36 49835675 IC50 = 0.5 nM T68290 C8O3UF 49835732 IC50 = 3 nM T68290 CU56CD 49862015 IC50 = 676 nM T68290 CMA62P 49862016 IC50 = 105 nM T68290 COY8Z0 49862017 IC50 = 3236 nM T68290 CEH26G 49862059 IC50 = 40 nM T68290 CEHY57 49862060 IC50 = 71 nM T68290 CI90VX 49862061 IC50 = 24 nM T68290 C6QN8X 49862100 IC50 = 12.6 nM T68290 CFB57Z 49862101 IC50 = 10 nM T68290 CCM26G 49862102 IC50 = 11 nM T68290 CDZL08 49862143 IC50 = 7.8 nM T68290 CVB95I 49862144 IC50 = 316 nM T68290 CWG62C 49862145 IC50 = 14.1 nM T68290 C37RZT 49862146 IC50 = 8.3 nM T68290 CGT50H 49862184 IC50 = 209 nM T68290 CO1Y6B 49862185 IC50 = 7.8 nM T68290 CJ0HY8 49862186 IC50 = 41 nM T68290 CD97QU 49862228 IC50 = 1.3 nM T68290 CXO39G 49862275 IC50 = 661 nM T68290 CKA53W 49862308 IC50 = 148 nM T68290 C8B2WE 49862309 IC50 = 174 nM T68290 CR13LF 49862310 IC50 = 447 nM T68290 C38BJK 49862365 IC50 = 83 nM T68290 C1Z9VQ 49862366 IC50 = 410 nM T68290 C6W1UJ 49862367 IC50 = 195 nM T68290 CIFP19 49862368 IC50 = 224 nM T68290 CMW23V 49862369 IC50 = 115 nM T68290 CI4J0A 49862370 IC50 = 200 nM T68290 C1XBM6 49862420 IC50 = 63 nM T68290 CKV06S 49862421 IC50 = 51 nM T68290 CN4GD6 49862422 IC50 = 1047 nM T68290 CA7K8Q 49862423 IC50 = 13 nM T68290 CS92IZ 49862471 IC50 = 10 nM T68290 C1NAQ5 49862472 IC50 = 15 nM T68290 C5OD6J 49862473 IC50 = 6 nM T68290 CFCH31 49862474 IC50 = 32 nM T68290 C29OGE 49862475 IC50 = 58 nM T68290 CU7T1N 49862476 IC50 = 60 nM T68290 CW36FO 49862535 IC50 = 23 nM T68290 CM94UQ 49862536 IC50 = 509 nM T68290 C69TUQ 49862719 IC50 = 29 nM T68290 CTQ19U 49862720 IC50 = 1660 nM T68290 CN6L9Y 49862793 IC50 = 1047 nM T68290 CN8PD3 49862794 IC50 = 339 nM T68290 CU3QE7 49862795 IC50 = 145 nM T68290 COA12C 49862796 IC50 = 200 nM T68290 C3N8YJ 49862797 IC50 = 63 nM T68290 CZPY13 49863204 IC50 = 4.5 nM T68290 C5GU2F 49863239 IC50 = 155 nM T68290 C18RNG 50925386 Ki = 140 nM T68290 C01DJG 50993971 Ki = 800 nM T68290 CW9X3R 50993972 Ki = 9.1 nM T68290 CIC7H1 50993973 Ki = 1.5 nM T68290 C3UB9Y 50993974 Ki = 0.83 nM T68290 CMS13V 50994055 Ki = 0.2 nM T68290 CPT6I5 50994056 Ki = 0.86 nM T68290 CB4X6Y 50994057 Ki = 0.16 nM T68290 CSY4W0 50994058 Ki = 0.2 nM T68290 CQ08HC 50994059 Ki = 0.17 nM T68290 C30WKN 50994060 Ki = 0.16 nM T68290 C8A1GN 50994137 Ki = 0.19 nM T68290 C6K3EJ 50994138 Ki = 0.32 nM T68290 CN6ZM0 50994139 Ki = 180 nM T68290 CF7SN9 50994140 Ki = 140 nM T68290 CU7M1P 50994141 Ki > 22000 nM T68290 C4FE0T 50994142 Ki = 0.15 nM T68290 CDC64G 52941172 IC50 > 10000 nM T68290 CJSD25 52941466 IC50 = 14.1 nM T68290 C71VFU 52941469 IC50 = 2.3 nM T68290 CBKG58 52941965 IC50 > 10000 nM T68290 CWB59N 52941968 IC50 = 18 nM T68290 CFP83K 52942699 IC50 = 10.5 nM T68290 CBM6K7 52942707 IC50 = 8.5 nM T68290 C12MHY 52942758 IC50 = 2.9 nM T68290 CW05MV 52942797 IC50 = 1.1 nM T68290 C8IC1X 52943191 IC50 > 10000 nM T68290 CQDG96 52943578 IC50 = 19.5 nM T68290 CMO15T 52944369 IC50 = 36 nM T68290 C9RY6V 52945164 IC50 = 11 nM T68290 C9B1ON 52946392 IC50 = 4.8 nM T68290 C5CJT3 52946393 IC50 = 1.1 nM T68290 CYL31K 52947479 IC50 = 692 nM T68290 C3PK2V 52948050 IC50 = 110 nM T68290 CD6CT7 52948442 IC50 = 2.3 nM T68290 CTV1C2 52948769 IC50 = 30.9 nM T68290 C75SHQ 52948860 IC50 = 1 nM T68290 CLIS74 52948911 IC50 = 31 nM T68290 C3TB7W 52949669 IC50 = 1.9 nM T68290 C56OCA 53317528 IC50 = 1584.89 nM T68290 C7I9AO 53317529 IC50 = 7943.28 nM T68290 CM60RJ 53317530 IC50 > 25118.86 nM T68290 C5A6IH 53317737 IC50 = 3981.07 nM T68290 C6FEH9 53318816 IC50 > 25118.86 nM T68290 CJAX07 53318817 IC50 = 15848.93 nM T68290 CG5AP6 53318818 IC50 = 15848.93 nM T68290 CJ3PN0 53319501 IC50 = 7.9 nM T68290 C7V2DA 53322116 IC50 = 13 nM T68290 CQ8O1R 53322117 IC50 = 27 nM T68290 C0QV5D 53322753 IC50 = 12589.25 nM T68290 CHB96K 53324300 IC50 = 1584.89 nM T68290 CR1L4Y 53325394 IC50 > 25118.86 nM T68290 CVU0J1 53326656 IC50 = 501.19 nM T68290 CWJB05 53364091 IC50 = 1.5 nM T68290 CT03IA 53377641 IC50 = 38 nM T68290 CX98BE 53377643 IC50 = 120 nM T68290 C7NC4V 53377644 IC50 = 0.5 nM T68290 C5WMZ4 53377646 IC50 = 3.5 nM T68290 C0G1HW 53377751 IC50 = 4000 nM T68290 COSL29 53377752 IC50 = 74 nM T68290 CTR8A5 53377864 IC50 = 8000 nM T68290 CR8U6P 53377865 IC50 > 20000 nM T68290 CDP97L 53377976 IC50 = 1.8 nM T68290 CW91VC 53378078 IC50 = 3.1 nM T68290 CI5OP3 53378080 IC50 = 5.6 nM T68290 C6CYR9 53378082 IC50 = 150 nM T68290 C1PDX9 53378184 IC50 = 310 nM T68290 C81RTV 53378188 IC50 = 3200 nM T68290 C1R7DL 53378291 IC50 = 110 nM T68290 C7BGP4 53378293 IC50 = 93 nM T68290 C5H3XK 53378295 IC50 = 1500 nM T68290 CPN6B8 53378493 IC50 = 0.7 nM T68290 CL40MU 53378494 IC50 = 5.2 nM T68290 CR2Y1U 53378704 IC50 = 8.8 nM T68290 CI63AX 53378705 IC50 = 13 nM T68290 CJ14TC 53378920 IC50 = 44 nM T68290 CAY12W 53378922 IC50 = 83 nM T68290 C2N6OY 53378924 IC50 = 17 nM T68290 CIJW35 53379043 IC50 = 2.2 nM T68290 C60DPQ 53379044 IC50 = 5.4 nM T68290 C1YH5J 53379045 IC50 = 5.7 nM T68290 CH1VR3 53379048 IC50 = 33 nM T68290 CF0WE8 53379159 IC50 = 88 nM T68290 CCT85S 53379268 IC50 = 10 nM T68290 CO32FE 53379269 IC50 = 93 nM T68290 C2Z4HC 53379270 IC50 = 160 nM T68290 C38RDM 53379272 IC50 = 15 nM T68290 CCG3S4 56666730 IC50 = 31.6 nM T68290 CK54CF 56670150 IC50 = 2.9 nM T68290 C69ILG 56670151 IC50 < 0.4 nM T68290 CA2Z0U 56676986 IC50 = 1.2 nM T68290 C24QMN 56680316 IC50 = 101 nM T68290 CX8M7Z 56683636 IC50 = 0.76 nM T68290 C1KR7M 56960717 IC50 = 12.4 nM T68290 C84CHB 57541268 IC50 > 4000 nM T68290 CH3M0B 59543520 IC50 = 13 nM T68290 CCR9Q8 59543629 IC50 = 0.3 nM T68290 C3ESJ1 59543757 IC50 = 0.8 nM T68290 CZV45P 59619390 IC50 = 26 nM T68290 CIM9F0 59780492 IC50 = 70 nM T68290 CXY2S6 59780538 IC50 = 790 nM T68290 CZ2FH1 59780570 IC50 = 70 nM T68290 CMTH79 59780582 IC50 = 260 nM T68290 CO6V9M 59780607 IC50 = 1750 nM T68290 CY46MU 59780611 IC50 = 2500 nM T68290 CK8MZ6 59780655 IC50 = 90 nM T68290 CPJ4W0 59780680 IC50 = 180 nM T68290 CLX2Y4 60148518 Ki = 33 nM T68290 C0DA6M 60166364 Ki = 40 nM T68290 C4G1SF 60166365 Ki = 45 nM T68290 COM7U3 60166366 Ki = 61 nM T68290 COQ82A 60166367 Ki = 60 nM T68290 C2Y7EK 60166492 Ki = 61 nM T68290 C4PHR1 60166493 Ki = 76 nM T68290 CG4DZ7 60166494 Ki = 200 nM T68290 C5E2PB 60166495 Ki = 94 nM T68290 CXD39V 60166496 Ki = 89 nM T68290 CM8XO5 60166497 Ki = 100 nM T68290 CA95CZ 60195809 IC50 = 3700 nM T68290 CY3VC4 60195810 IC50 = 2110 nM T68290 CVRJ91 60195812 IC50 = 515 nM T68290 CE6AH0 60195813 IC50 = 2070 nM T68290 C8ILH6 60195902 IC50 = 1030 nM T68290 CX4N2V 60195903 IC50 = 3360 nM T68290 C4PQ6E 60195904 IC50 > 100000 nM T68290 CNUI89 60195905 IC50 > 70000 nM T68290 C23JUZ 60195906 IC50 > 100000 nM T68290 CDA2M1 66995873 Ki > 10000 nM T68290 C85OHR 67475270 IC50 = 7.7 nM T68290 CUI42K 69098820 IC50 = 10 nM T68290 CJ8VZ4 69098861 IC50 = 1630 nM T68290 CRZJ37 69098878 IC50 = 30 nM T68290 C9W4KR 69098883 IC50 = 70 nM T68290 CTZC78 69099077 IC50 = 160 nM T68290 C1MI4Q 69099090 IC50 = 120 nM T68290 CX21VM 69099137 IC50 = 100 nM T68290 CTP1B4 69108181 IC50 = 630 nM T68290 CHR0T8 69319709 IC50 = 40 nM T68290 C6K5PZ 69320181 IC50 = 40 nM T68290 CWLK73 69320228 IC50 = 30 nM T68290 CC3E5A 69322125 IC50 = 120 nM T68290 C67VLI 69322366 IC50 = 60 nM T68290 CJFU46 69323931 IC50 = 4560 nM T68290 C7A6DR 69324191 IC50 = 30 nM T68290 CJ4E7Y 69924515 IC50 = 49 nM T68290 CM7C2P 69924681 IC50 = 760 nM T68290 CD21FS 69924711 IC50 = 2 nM T68290 C4JPF2 69924862 IC50 = 0.1 nM T68290 C90POH 69924990 IC50 = 110 nM T68290 CBR31D 69925026 IC50 = 1.1 nM T68290 CJ3C8F 69925113 IC50 = 93 nM T68290 CS8E0W 69925136 IC50 = 18 nM T68290 CDE6I0 69925138 IC50 = 15 nM T68290 C9RMC7 69925195 IC50 = 72 nM T68290 CDE2Z8 69925409 IC50 = 3.2 nM T68290 C1MAX3 69925414 IC50 = 110 nM T68290 C9SQC3 69925439 IC50 = 39 nM T68290 C7N2QL 69925473 IC50 = 4.2 nM T68290 CWT67K 69925480 IC50 = 61 nM T68290 CEH9V1 69925506 IC50 = 13 nM T68290 CVJ5F3 69925527 IC50 = 2.3 nM T68290 CU3R2L 69925600 IC50 = 46 nM T68290 C0DO9E 69925672 IC50 = 210 nM T68290 C4PNI0 69925805 IC50 = 5.9 nM T68290 C95HQC 69925936 IC50 = 39 nM T68290 CKFG50 69926162 IC50 = 130 nM T68290 CSF35K 70274227 IC50 = 549 nM T68290 CI0XF8 70274815 IC50 = 3981.07 nM T68290 CXT5G7 70275845 IC50 = 1510 nM T68290 C5P3BO 70275923 IC50 > 11800 nM T68290 CCG16F 70276365 IC50 = 1584.89 nM T68290 C0T3LC 70276605 IC50 = 2290 nM T68290 CE1J0O 70276811 IC50 = 1995.26 nM T68290 C06WFN 70276830 IC50 > 10000 nM T68290 CDQ85E 70276990 IC50 > 100000 nM T68290 CGET13 70278898 IC50 = 1258.93 nM T68290 C2GT5H 70280758 IC50 = 2511.89 nM T68290 CI53XU 70281040 IC50 = 3750 nM T68290 CA6DM2 70281073 IC50 = 1584.89 nM T68290 CZ84UX 70682584 IC50 > 1995.26 nM T68290 CL9RE3 70686820 IC50 = 3162.28 nM T68290 C65EDY 70686822 IC50 > 2511.89 nM T68290 C5IYR0 70688897 IC50 = 2511.89 nM T68290 CZOF81 70693115 IC50 = 1584.89 nM T68290 CMFW03 70693116 IC50 = 1584.89 nM T68290 C5RSJ0 70693117 IC50 = 1584.89 nM T68290 C01IDC 70695171 IC50 > 2511.89 nM T68290 C34WHG 70697225 IC50 = 3162.28 nM T68290 CUB38S 71449749 IC50 > 4000 nM T68290 CS60PU 71450699 IC50 = 1.6 nM T68290 CS58YC 71450700 IC50 = 3 nM T68290 C61VTL 71450701 IC50 = 1 nM T68290 C08LGJ 71451733 IC50 = 1680 nM T68290 CI7Z8B 71451734 IC50 = 1150 nM T68290 C2UN6D 71452029 IC50 > 100000 nM T68290 CG8T7Z 71452030 IC50 > 100000 nM T68290 C2KR7V 71452494 IC50 = 4 nM T68290 C9C2KR 71452495 IC50 = 8.8 nM T68290 C4PQ9H 71452496 IC50 = 23 nM T68290 C57CDN 71452524 IC50 = 150 nM T68290 CN4B9F 71452525 IC50 = 400 nM T68290 C2OGP1 71453559 IC50 = 2600 nM T68290 CDR10X 71453560 IC50 = 2260 nM T68290 CPGT63 71454020 Ki = 8400 nM T68290 CZ6M8U 71454284 IC50 = 0.3 nM T68290 CP7H6S 71454285 IC50 = 20 nM T68290 CAT5O1 71454286 IC50 = 4.6 nM T68290 CFUS41 71455276 IC50 = 1290 nM T68290 CUQL74 71455277 IC50 = 1750 nM T68290 C0KUW5 71455278 IC50 = 1100 nM T68290 C7Z0HF 71455279 IC50 = 1300 nM T68290 C78BKL 71455561 IC50 > 100000 nM T68290 CU48QH 71455759 Ki = 6600 nM T68290 C9YJG7 71457065 IC50 = 1090 nM T68290 CLD37I 71457817 IC50 = 4.9 nM T68290 C3IH8Z 71457841 IC50 = 13 nM T68290 CCH47M 71458921 IC50 = 2950 nM T68290 CP7MZ5 71458922 IC50 = 1230 nM T68290 CCA46N 71458923 IC50 = 1450 nM T68290 CQT1C2 71458924 IC50 = 1220 nM T68290 C6RZF3 71459429 Ki = 750 nM T68290 CF69OZ 71459754 IC50 = 0.6 nM T68290 CE9LP1 71460574 IC50 = 258 nM T68290 CDW0I7 71460731 IC50 = 1050 nM T68290 CL6Y4C 71460733 IC50 = 807 nM T68290 CKB60I 71461472 IC50 = 27 nM T68290 C8XW0G 71461473 IC50 = 93 nM T68290 C18KJW 71463174 IC50 = 28 nM T68290 C0JFQ2 71463175 IC50 = 29 nM T68290 C7GX8H 71463202 IC50 = 0.6 nM T68290 CPT0L4 71553088 IC50 = 60 nM T68290 CCF5Q2 71553157 IC50 = 100 nM T68290 CER82H 71612695 Ki = 28000 nM T68290 CL0JD4 71624114 IC50 > 1000 nM T68290 C5NV8E 71624115 IC50 = 3 nM T68290 C37RTB 71624116 IC50 = 3.1 nM T68290 C2U0OH 71624117 IC50 = 2.4 nM T68290 C8DZ6U 71624118 IC50 = 3.3 nM T68290 CQ0Z5J 71624239 IC50 = 2.7 nM T68290 C3L0HN 71624240 IC50 = 3.3 nM T68290 CFDY38 71624241 IC50 = 3.7 nM T68290 CLF8R4 71624242 IC50 = 3.3 nM T68290 CL2Z8C 71624243 IC50 = 3.5 nM T68290 C8SGK6 71624246 IC50 = 3.3 nM T68290 CP0D4W 71624247 IC50 = 4.3 nM T68290 CJ93QW 71624361 IC50 = 2 nM T68290 CM64QD 71624362 IC50 = 1.1 nM T68290 CK64NT 71624363 IC50 = 4.1 nM T68290 CRMY89 71624364 IC50 = 2.3 nM T68290 CZM2V4 71624365 IC50 = 3.2 nM T68290 CYZI36 71624480 IC50 = 3.2 nM T68290 CNVW79 71624481 IC50 > 100 nM T68290 CW6Q4D 71624482 IC50 = 18.1 nM T68290 CS10EX 71624483 IC50 = 24.6 nM T68290 C6U4CM 71624484 IC50 > 100 nM T68290 CDM4O5 71624594 IC50 = 36.6 nM T68290 C6R7FN 71625894 IC50 = 3.5 nM T68290 CR8GE0 71625895 IC50 = 45.4 nM T68290 C81CSV 71625896 IC50 = 12.4 nM T68290 C3IV4B 71625897 IC50 = 20.7 nM T68290 C40MTY 71625898 IC50 = 83.7 nM T68290 CAN6X5 71656574 IC50 = 2700 nM T68290 CU32JC 71717327 IC50 = 110 nM T68290 CSN07F 72793721 IC50 = 271 nM T68290 C6I4RC 72793722 IC50 = 12 nM T68290 CO1W8E 72793723 IC50 = 18 nM T68290 CY1IU2 73345852 Ki = 20000 nM T68290 COJN04 73347330 IC50 = 3.3 nM T68290 C5AMR2 73348056 IC50 > 100000 nM T68290 CJQE58 73348851 Ki = 56000 nM T68290 C31JUR 73348857 Ki = 8500 nM T68290 C95BEA 73348858 Ki = 41100 nM T68290 CAYM96 73351955 Ki = 12000 nM T68290 CY9JN7 73353390 IC50 = 156 nM T68290 CJ6CQ1 73356205 Ki = 290 nM T68290 C0ZDB4 76313697 IC50 = 640 nM T68290 CX26GW 76328142 IC50 = 830 nM T68290 C62SML 90655967 IC50 > 10000 nM T68290 CJ7LT3 90655968 IC50 > 10000 nM T68290 CB61WC 90655969 IC50 > 10000 nM T68290 CIS56R 90663177 Ki = 5.9 nM T68290 CU71EO 90663180 Ki = 11 nM T68290 CX37IK 90663181 Ki = 1.8 nM T68290 CH68BZ 91885514 Ki = 5000 nM T68290 C8E4WS 102323332 IC50 > 50000 nM T68290 CVJF59 118716317 Ki = 0.777 nM T68290 CA79YF 118716318 Ki = 0.176 nM T68290 C3Q5BM 118716319 Ki = 0.13 nM T68290 CI6H0V 118716320 Ki = 793 nM T68290 CL4ES1 118716560 IC50 = 1170 nM T68290 CZF4T5 118716561 IC50 = 1290 nM T68290 C3ZE5A 118716562 IC50 = 4000 nM T68290 CTE34I 118720232 IC50 > 100000 nM T68290 CSD62B 118720233 IC50 > 100000 nM T68290 C9WF7Q 118720234 IC50 = 1000 nM T68290 C76HIO 118720235 IC50 = 24000 nM T68290 CAT1R6 118720236 IC50 > 100000 nM T68290 CGAF42 118720237 IC50 > 100000 nM T68290 CJ28KZ 118720238 IC50 > 100000 nM T68290 CPH2V9 118720239 IC50 > 100000 nM T68290 CCXD81 122186478 Ki = 4000 nM T68290 C3C7BJ 122186482 Ki = 1000 nM T68290 CV04JO 127037715 IC50 > 50000 nM T68290 CJ27CG 127042051 IC50 > 50000 nM T68290 CAT46D 127042341 IC50 > 50000 nM T68290 CMT2B9 127049869 Ki = 2250 nM T68290 C43APM 127050163 Ki = 1000 nM T68290 C8VKA5 127050164 Ki = 490 nM T68290 CZ54XC 127050165 Ki = 186 nM T68290 CI2C3V 127050166 Ki = 352 nM T68290 C7V8XZ 127051317 Ki = 1800 nM T68290 CSK16Q 127051318 Ki = 4230 nM T68290 C7YI4M 127051342 Ki = 180 nM T68290 C6NFU9 127051343 Ki = 178 nM T68290 C6SD7P 127051344 Ki = 2660 nM T68290 CY5CV6 127051345 Ki = 4480 nM T68290 C2CT4O 134134083 IC50 = 23 nM T68290 CX7UT0 134135239 IC50 = 23 nM T68290 COU6A4 134135795 IC50 = 23 nM T68290 CD0UE9 134136855 IC50 = 17 nM T68290 CF8VA4 134138144 IC50 = 17 nM T68290 CFE54U 134139713 IC50 = 23 nM T68290 C3PEW2 134141970 IC50 = 90 nM T68290 CV36BU 134142724 IC50 = 136 nM T68290 C4BXO1 134144535 IC50 = 28 nM T68290 CE8Q2J 134147121 IC50 = 23 nM T68290 C8WYF6 134147241 IC50 = 102 nM T68290 C0YG8C 134148335 IC50 = 17 nM T68290 C7CH0G 134151560 IC50 = 23 nM T68290 C4TS3J 134154893 IC50 = 23 nM T68290 CTQY96 136117851 IC50 = 9 nM T68290 CM4ZW3 137651124 Ki = 7260 nM T68290 CFQ25D 145967499 IC50 = 710 nM T68290 CIVB10 145967715 IC50 = 1 nM T68290 CLI6T0 145967952 IC50 = 195 nM T68290 CC4AG7 145968405 IC50 > 5000 nM T68290 CDS31M 145968622 IC50 = 85 nM T68290 CA40YU 145969275 IC50 = 283 nM T68290 CB0Y7Z 145969438 IC50 > 5000 nM T68290 C2WCK0 145969450 IC50 = 3583 nM T68290 CL7KO9 145969878 IC50 = 2371 nM T68290 C3NAS7 145970030 IC50 > 5000 nM T68290 CS08XI 145970918 IC50 > 5000 nM T68290 C9XKW2 145970931 IC50 = 253 nM T68290 CXW3F1 145982578 IC50 = 400 nM T68290 CY7XE4 145982644 IC50 = 30 nM T68290 C56AXR 145982654 IC50 = 20 nM T68290 C7S2TX 145983004 IC50 = 200 nM T68290 C7V2ZF 145983823 IC50 = 20 nM T68290 CV1A6D 145983891 Ki = 2 nM T68290 CV8HP6 145984203 Ki = 30 nM T68290 C3JIQ4 145984217 IC50 = 100 nM T68290 CT8QM9 145984597 IC50 = 300 nM T68290 CJM6L4 145984752 IC50 = 50 nM T68290 C0BC2Z 145984777 IC50 = 20 nM T68290 CGC54P 145985016 IC50 = 200 nM T68290 C2LB8K 145985094 IC50 = 20 nM T68290 CNT63X 145985191 IC50 = 10 nM T68290 CX6JT1 145985564 IC50 = 200 nM T68290 CJE7L9 145985615 IC50 = 800 nM T68290 CL2B3Y 145985677 IC50 = 10 nM T68290 CQ2RS8 145986120 IC50 = 80 nM T68290 CM53FT 145986712 Ki = 17 nM T68290 CRD65W 145987430 Ki = 15000 nM T68290 COZ6P5 145987960 IC50 = 190 nM T68290 C7ZCW3 145988622 IC50 = 18 nM T68290 C9OAK6 145989037 IC50 = 1.1 nM T68290 C87GKT 145989707 IC50 = 382 nM T68290 CUAY08 148018738 IC50 > 10000 nM T68290 CQK39B 149491764 IC50 > 10000 nM T68290 C1ZX5D 149494192 IC50 > 10000 nM T68290 CKT12D 155510715 Ki = 1410 nM T68290 CO2Y0C 155523098 Ki = 870 nM T68290 CBN12I 155524050 Ki = 735 nM T68290 CO3ZF7 155541809 Ki = 320 nM T68290 CXYT09 155551122 Ki = 239 nM T68290 CCF86H 155553085 Ki = 1800 nM T68290 C6O9FK 155556968 Ki = 370 nM T68290 C58OLD 44517711 IC50 = 199.53 nM T68290 CT3S1I 44517712 IC50 = 63.1 nM T68290 CFT38D 45267632 IC50 = 316.23 nM T68290 COU83P 45267640 IC50 = 2.512 nM T68290 C1U4IF 45267645 IC50 = 316.23 nM T68290 CDG5S8 45268499 IC50 = 100 nM T68290 CV8PZ3 45268510 IC50 = 794.33 nM T68290 C89ADF 45269361 IC50 = 79.43 nM T68290 C58PZI 45269375 IC50 = 19.95 nM T68290 C5O9EF 45270206 IC50 = 15.85 nM T68290 C07ADH 45270207 IC50 = 79.43 nM T68290 CVGE81 45270212 IC50 = 63.1 nM T68290 C78EXG 45271021 IC50 = 125.89 nM T68290 C5MBC4 45271038 IC50 = 79.43 nM T68290 C65QLD 45271887 IC50 = 316.23 nM T68290 CIL8O6 45271888 IC50 = 316.23 nM T68290 CLFD35 45272742 IC50 = 316.23 nM T68290 C3WF8S 45272748 IC50 = 630.96 nM T68290 CQO98K 45272752 IC50 = 7.943 nM T68290 C9A0IH 45272753 IC50 = 63.1 nM T68290 CSYU09 45273681 IC50 = 251.19 nM T68290 D00FGA 73737 IC50 = 25118.86 nM T68290 D01IFO 49863205 IC50 = 2884 nM T68290 D01JGB 46881498 IC50 = 2239 nM T68290 D01NCW 11534772 IC50 = 9000 nM T68290 D01YNC 23648531 Ki = 4100 nM T68290 D02FPU 52945617 IC50 = 1070 nM T68290 D04BGT 46881451 IC50 = 950 nM T68290 D05MDE 11505372 IC50 = 13000 nM T68290 D05VEV 11556056 IC50 = 6900 nM T68290 D05WZF 10129151 IC50 = 130 nM T68290 D06NEB 11693148 IC50 = 150 nM T68290 D06VIP 14774521 Ki = 6200 nM T68290 D06WQP 60148519 Ki = 0.55 nM T68290 D07FLB 11637576 Ki = 550 nM T68290 D07RSA 11696652 Ki = 240 nM T68290 D07SOQ 11652399 Ki = 2500 nM T68290 D08TMM 9851116 IC50 = 0.6 nM T68290 D09AHN 11492732 Ki = 130 nM T68290 D09FGQ 123985 IC50 = 7 nM T68290 D09GZQ 11713852 IC50 = 12000 nM T68290 D09IMK 11621748 IC50 = 3300 nM T68290 D0A5WN 11621347 IC50 = 67000 nM T68290 D0A7ER 11514386 Ki = 900 nM T68290 D0A8OV 11086036 Ki = 1400 nM T68290 D0B2FE 46882093 IC50 > 10000 nM T68290 D0B3US 11585523 IC50 = 13000 nM T68290 D0D0LD 9913088 IC50 = 95 nM T68290 D0G8OD 11702208 Ki = 130 nM T68290 D0I0MU 11534625 IC50 = 700 nM T68290 D0JF8D 11551481 Ki = 970 nM T68290 D0JN8Q 11702265 Ki = 77 nM T68290 D0K0KT 11621207 IC50 = 3000 nM T68290 D0L9VP 5287864 Ki < 0.1 nM T68290 D0QY3R 11513217 IC50 = 7100 nM T68290 D0RL4S 11714476 IC50 = 10000 nM T68290 D0U0XG 11709032 Ki = 660 nM T68290 D0U4TY 11694425 IC50 = 1300 nM T68290 D0V5LJ 10168449 IC50 = 100 nM T68290 D0Y5IQ 44255320 IC50 = 10000 nM T68290 D0Y5LX 11622731 IC50 > 10000 nM T68290 D0Z0PR 9912381 Ki = 47000 nM T50547 D04ZIJ 5478883 IC50 = 0.9 nM T50547 C2AX7O 445304 Ki = 25 nM T50547 CPS5Z7 6539218 Ki = 16 nM T50547 CV5K3I 6539219 Ki = 27 nM T50547 C7UR8H 6539220 Ki = 5.4 nM T50547 CYA9X5 6539221 Ki = 0.5 nM T50547 CY6M5W 6539222 Ki = 5.4 nM T50547 CEX3D8 6539224 Ki = 49 nM T50547 C9DOI1 6539225 Ki = 6.7 nM T50547 CR7A3L 6539226 Ki = 8.9 nM T50547 C0H5ZW 6539227 Ki = 4.1 nM T50547 CUQ6T5 6539228 Ki = 53 nM T50547 C32QNI 6539229 Ki = 8.1 nM T50547 CZN02I 6539230 Ki = 6.4 nM T50547 CXPO09 6539231 Ki = 32 nM T50547 C4GX1T 6539232 Ki = 3.4 nM T50547 C2YKM3 6539233 Ki = 57 nM T50547 COLZ28 6539234 Ki = 40 nM T50547 CJ14EB 6539235 Ki = 24 nM T50547 CQ5O9H 6539236 Ki = 29 nM T50547 CIY71M 6539237 Ki = 59 nM T50547 CIWC50 6539238 Ki = 619 nM T50547 C9VQZ4 6539239 Ki = 822 nM T50547 C4AXO5 6539241 Ki = 163 nM T50547 CY8HL5 6539242 Ki > 1500 nM T50547 CA78BY 6539243 Ki = 27 nM T50547 CB2O4C 6539244 Ki = 1.4 nM T50547 CEX54J 6539245 Ki = 2.5 nM T50547 C61TOP 6539246 Ki = 5.8 nM T50547 C01MAJ 6539247 Ki = 0.8 nM T50547 CV7NB4 6539248 Ki = 8.4 nM T50547 CMHE43 6539249 Ki = 0.5 nM T50547 CQO6I0 6539250 Ki = 1.3 nM T50547 CHC57F 6539251 Ki = 23 nM T50547 CT30RS 6539252 Ki = 4.4 nM T50547 CNZ8E9 6539253 Ki = 3.7 nM T50547 CV9Q8Z 6539254 Ki = 7.2 nM T50547 C3VB5A 6539255 Ki = 37 nM T50547 C6H5IQ 6539256 Ki = 32 nM T50547 CF30BP 6539257 Ki = 2.6 nM T50547 CZ40TI 6539258 Ki > 2000 nM T50547 C3WI4Y 6539261 Ki > 2000 nM T50547 CE51XA 6539262 Ki ~ 2900 nM T50547 CN6OX1 6539263 Ki > 2000 nM T50547 CB89QP 6539264 Ki ~ 2100 nM T50547 CB14ZY 6539265 Ki ~ 8000 nM T50547 CBF54P 6539266 Ki = 98 nM T50547 CM6X7H 6539267 Ki = 68 nM T50547 C6RQ9Z 6539268 Ki = 115 nM T50547 C0Y9GC 6539269 Ki = 63 nM T50547 CWIJ07 6539270 Ki = 437 nM T50547 CSD6R5 6539271 Ki = 1300 nM T50547 CWR7C9 6539272 Ki = 469 nM T50547 CXT20F 6539273 Ki = 1100 nM T50547 CURY46 6539274 Ki = 1000 nM T50547 CLE4I2 6539275 Ki = 530 nM T50547 C1SUG3 6539276 Ki > 2000 nM T50547 CV2JK1 6539277 Ki = 2046 nM T50547 C0J2NU 11204230 Ki = 116 nM T50547 C1YFZ0 11214849 IC50 = 1123 nM T50547 CEDP95 11215989 Ki = 2.1 nM T50547 CENB36 11227366 Ki = 2.7 nM T50547 CE1B6S 11239445 Ki = 3.3 nM T50547 CX30NP 11249866 Ki = 188 nM T50547 CZ4X0A 11250844 Ki = 5.9 nM T50547 C8PHK2 11273154 Ki = 1.9 nM T50547 C5ZDP8 11284770 IC50 = 1162 nM T50547 C2C4XA 11285489 Ki = 0.3 nM T50547 C4BHV0 11285517 Ki = 0.4 nM T50547 C98FEY 11285691 Ki > 3000 nM T50547 C5BO7P 11296167 Ki = 1 nM T50547 C2QK0E 11308017 Ki = 221 nM T50547 C1RG5P 11399816 Ki = 0.7 nM T50547 C6UT8Z 11399839 Ki = 0.3 nM T50547 CSJD04 11410402 Ki = 278 nM T50547 C9YKP7 11505733 Ki > 3000 nM T50547 CJ9NL1 11505900 Ki > 3000 nM T50547 C1VEC2 11513333 Ki = 19 nM T50547 C8P5JQ 11513415 Ki = 1090 nM T50547 CF2JU9 11520423 Ki > 3000 nM T50547 C6U9JR 11527693 Ki = 261 nM T50547 CKU80T 11534178 Ki > 3000 nM T50547 CKY5C8 11534582 Ki > 3000 nM T50547 CS0H9X 11534953 Ki > 3000 nM T50547 C02DGS 11541427 Ki = 124 nM T50547 C8SFN6 11541810 Ki > 3000 nM T50547 CB59KM 11564069 Ki = 38 nM T50547 C8RPH4 11607313 Ki = 9 nM T50547 C7XU9H 11614671 Ki = 2000 nM T50547 CSR87I 11629093 Ki = 1600 nM T50547 CN9AO7 11636216 Ki = 31 nM T50547 CA45GE 11657449 Ki = 698 nM T50547 CHXL54 11664893 Ki = 11 nM T50547 CM46HF 11671674 IC50 = 123 nM T50547 CXN6V9 11685086 Ki > 3000 nM T50547 CWTA90 11707562 Ki = 198 nM T50547 CIDF31 11721953 Ki = 6 nM T50547 CH1Y8K 11764107 Ki = 0.4 nM T50547 CD1N7A 11787369 Ki = 1 nM T50547 COIH49 16121203 Ki = 74 nM T50547 CY91SZ 44341490 Ki = 3.9 nM T50547 C0HF9G 44418735 Ki = 765 nM T50547 CE7TW9 44418736 Ki = 81 nM T50547 C2LIW7 44418737 Ki = 58 nM T50547 C6OI8E 44418738 Ki = 11 nM T50547 C93HCD 44418739 Ki = 17 nM T50547 CW1NU7 44418740 Ki = 33 nM T50547 CF6PJ1 44418741 Ki = 1 nM T50547 CY6U5Q 44418742 Ki = 230 nM T50547 C7AFS5 44527662 IC50 = 700 nM T50547 CM0A8K 44532986 IC50 = 18000 nM T50547 CW6V8G 45267698 IC50 = 16545 nM T50547 C1UN6X 45268565 IC50 > 25000 nM T50547 C86LOA 45268566 IC50 = 4391 nM T50547 CBA06Z 45268568 IC50 > 25000 nM T50547 CKF16D 45271072 IC50 > 25000 nM T50547 C8GB5K 45272786 IC50 = 2642 nM T50547 CT6W4D 45273746 IC50 > 25000 nM T50547 C3X0EZ 59688843 IC50 = 104 nM T50547 CM9FX0 59688861 IC50 = 113 nM T50547 C5DTE9 71520763 IC50 = 3100 nM T50547 C1BY0I 85470144 IC50 = 4600 nM T50547 CSM4C1 86288475 IC50 = 300 nM T50547 CV51KR 86288476 IC50 = 250 nM T50547 CS7ZM6 90655842 IC50 = 470 nM T50547 CQK42C 90655843 IC50 = 600 nM T50547 C64ASN 90655844 IC50 = 330 nM T50547 C65BUL 90655845 IC50 = 6100 nM T50547 COG5V7 90655846 IC50 = 750 nM T50547 CL81MW 90655847 IC50 = 1600 nM T50547 CAC0H4 90655848 IC50 = 7600 nM T50547 CYS25V 90655849 IC50 = 200 nM T50547 CH9VJ1 90655850 IC50 = 430 nM T50547 CYV70Z 90655851 IC50 = 18000 nM T50547 CPGK89 90655852 IC50 = 2300 nM T50547 C48HVL 90655853 IC50 = 45000 nM T50547 C4FR5P 90655854 IC50 = 360 nM T50547 C2GR6X 90655855 IC50 = 380 nM T50547 CL07NM 90655856 IC50 = 4100 nM T50547 CXAP16 90655857 IC50 = 350 nM T50547 CY19SM 90664068 Ki = 727 nM T50547 CZK0L7 105539825 IC50 = 1200 nM T50547 C2XHZ8 127026505 IC50 = 6000 nM T50547 CB3X2O 127026506 IC50 = 2400 nM T50547 C3DIN6 127027428 IC50 = 2300 nM T50547 CJM2K9 127027429 IC50 = 3700 nM T50547 C9RKY8 127027430 IC50 = 2000 nM T50547 C5XU8O 127027434 IC50 = 300 nM T50547 C51ONW 127027435 IC50 = 300 nM T50547 CZ0M8K 127027436 IC50 = 800 nM T50547 CR36NE 127027761 IC50 = 270 nM T50547 CHBD07 127027762 IC50 = 500 nM T50547 C7ZI6Q 127028384 IC50 = 9400 nM T50547 C7W8FM 127028385 IC50 = 480 nM T50547 C2E3QR 127028386 IC50 = 1400 nM T50547 C9H3QY 127028711 IC50 = 2000 nM T50547 C5CR4Z 127028712 IC50 = 3200 nM T50547 CLGB70 127038526 IC50 = 52000 nM T50547 CAT8G7 127039677 IC50 = 6500 nM T50547 C9LAO0 127040014 IC50 = 36000 nM T50547 CSC48Q 145968177 IC50 = 740 nM T50547 C24PUM 145968574 IC50 = 16700 nM T50547 CJ2V6B 145968904 IC50 = 2000 nM T50547 C8DOU5 145968976 IC50 = 1000 nM T50547 C1D6MG 145969118 IC50 = 700 nM T50547 CT1V0I 145969327 IC50 = 3000 nM T50547 CYH45E 145970255 IC50 = 5000 nM T50547 CVAW24 145970337 IC50 = 20 nM T50547 CT57RL 145970338 IC50 = 80 nM T50547 CDR2G9 145970368 IC50 = 90 nM T50547 CM8X7O 145970397 IC50 = 600 nM T50547 CP8A0Z 145970407 IC50 = 2400 nM T50547 C4F6NT 145970582 IC50 = 11500 nM T50547 CH9P3X 145970804 IC50 = 3500 nM T50547 CZ3X4R 145970818 IC50 = 1300 nM T50547 CS64YI 145970835 IC50 = 50 nM T50547 C95VSG 145987742 IC50 = 3400 nM T50547 C5PA1C 145988827 IC50 = 1000 nM T50547 C8XOC6 155511155 IC50 = 2000 nM T50547 CW89FM 155520640 IC50 = 1100 nM T50547 C85GWP 155521302 IC50 = 780 nM T50547 COG6S8 155524310 IC50 = 2500 nM T50547 CTKF74 155530540 IC50 = 5600 nM T50547 CRN6V8 155537831 IC50 = 800 nM T50547 C03KZX 155539456 IC50 = 2000 nM T50547 CVBR73 155539645 IC50 = 7400 nM T50547 CJB9K1 155540162 IC50 = 280 nM T50547 C25CXT 155542250 IC50 = 10300 nM T50547 CMN6E1 155556535 IC50 = 1800 nM T50547 C7DH9B 155556912 IC50 = 100 nM T50547 D06BKP 44342336 IC50 = 500 nM T50547 D08AES 11578664 Ki = 1837 nM T50547 D0S3BO 9895503 IC50 = 280 nM T50547 D0S4BV 657149 IC50 = 655 nM T99685 D06OMK 445643 IC50 = 3.162 nM T99685 D09XZB 123631 IC50 > 50000 nM T99685 D0B3HD 2519 IC50 = 400000 nM T99685 D0E6XR 3062316 IC50 = 35000 nM T99685 D0ES1Q 6918289 IC50 = 1760 nM T99685 D0J5VR 11625818 IC50 > 1000 nM T99685 D0R0MW 5329102 IC50 > 50000 nM T99685 D0S5LD 135565596 IC50 = 45 nM T99685 D0V7WS 9876378 IC50 = 3.3 nM T99685 D0W5HK 216239 IC50 > 50000 nM T99685 D01PGR 16123056 IC50 = 157 nM T99685 D01QSO 16654980 IC50 = 94 nM T99685 D03DPZ 45375953 Ki = 1 nM T99685 D03EZE 25167777 IC50 = 0.31 nM T99685 D03LWG 53235510 IC50 > 10000 nM T99685 D03XAQ 49784945 IC50 = 1600 nM T99685 D05EXN 58298316 IC50 = 10 nM T99685 D07BGC 57384863 Ki = 70 nM T99685 D07EHV 44814409 IC50 > 9100 nM T99685 D08QGT 17755052 IC50 = 3 nM T99685 D0AW5T 9849735 IC50 = 3100 nM T99685 D0D8JB 44516953 IC50 = 0.4 nM T99685 D0E6UZ 54575456 IC50 = 431 nM T99685 D0H9DA 54761306 IC50 = 370 nM T99685 D0N5JZ 25033539 IC50 = 7.9 nM T99685 D0O1IM 58298318 IC50 = 21 nM T99685 D0O1LD 11647372 IC50 = 350 nM T99685 D0O6VZ 25254071 Ki = 17 nM T99685 D0TU7B 58507717 Ki = 62 nM T99685 D0U8QH 59239165 Ki = 3.8 nM T99685 D0UP1Z 51001932 Ki = 1200 nM T99685 D0VG0D 11977753 IC50 = 5 nM T99685 D0W7HE 56649450 IC50 > 9100 nM T99685 D0XD4I 118502708 IC50 = 200 nM T99685 D0Z2UQ 25262792 IC50 = 2.8 nM T99685 D04PGB 445501 IC50 = 20892.96 nM T99685 D05HIJ 135565159 IC50 > 10000 nM T99685 D09SFV 3973 IC50 = 2500 nM T99685 D0K1VK 25262965 IC50 = 4 nM T99685 D0P1JI 312145 IC50 = 40 nM T99685 D0U2TQ 644215 IC50 = 800 nM T99685 CB1VW3 1400 IC50 = 9318 nM T99685 CH5QF8 1018277 IC50 = 570 nM T99685 CRGP15 1420707 IC50 = 52200 nM T99685 CT2VP9 1471775 IC50 = 1410 nM T99685 C9LG0N 1476679 IC50 = 5000 nM T99685 C49EKU 1862374 IC50 = 8300 nM T99685 C0NMD8 1882360 IC50 = 57600 nM T99685 C7CSH6 2024268 IC50 = 32200 nM T99685 CQ02GR 2930286 IC50 = 54100 nM T99685 C6T0BZ 4899677 IC50 = 20400 nM T99685 C4G6WY 5253082 IC50 > 2000 nM T99685 CZ7GL8 9809998 IC50 = 9.6 nM T99685 CNQJ46 9867340 IC50 = 193 nM T99685 CJ79RC 9879653 IC50 = 37 nM T99685 C7HMO6 11526786 IC50 = 2920 nM T99685 CFZO21 11979157 IC50 = 2 nM T99685 CBZU35 11997784 IC50 = 460 nM T99685 CEBI25 12050235 IC50 < 10000 nM T99685 CJCG06 12050236 IC50 < 10000 nM T99685 C0KX2Q 12050237 IC50 < 10000 nM T99685 C2DS5Z 12050238 IC50 < 10000 nM T99685 C63PLZ 12050239 IC50 < 10000 nM T99685 CZ7UR5 12050240 IC50 < 10000 nM T99685 CV9US5 16736978 IC50 = 3 nM T99685 C59CVU 19689599 IC50 > 20000 nM T99685 CTF23G 20644743 IC50 > 50000 nM T99685 CZ7V8L 21048651 IC50 > 50000 nM T99685 C0EJK3 23585071 IC50 = 288.4 nM T99685 CEYL29 23585510 IC50 > 9100 nM T99685 CBL37C 23642173 IC50 > 9100 nM T99685 C0EKO5 24772654 IC50 > 10000 nM T99685 CBS5J4 24804985 IC50 = 28 nM T99685 C9PA0M 24807809 IC50 = 28600 nM T99685 C5E4QN 24807810 IC50 > 20000 nM T99685 C3QKS1 24807976 IC50 = 5600 nM T99685 CGJ60P 24807978 IC50 = 14000 nM T99685 CIPF03 24808145 IC50 > 20000 nM T99685 C2XLC5 24808146 IC50 > 20000 nM T99685 C7DX6N 24808147 IC50 = 6500 nM T99685 CY61FQ 24808148 IC50 = 8700 nM T99685 C72QHP 24808149 IC50 > 20000 nM T99685 CBMA95 24808336 IC50 > 20000 nM T99685 C7FD1B 24808337 IC50 > 20000 nM T99685 CCP2M3 24822704 IC50 > 50000 nM T99685 CB79YC 24905143 IC50 = 2100 nM T99685 C2DC9J 24905144 IC50 = 100000 nM T99685 CN6V8Z 24905145 IC50 = 72 nM T99685 CSB7P5 24905148 IC50 = 4800 nM T99685 CGSF21 24905149 IC50 = 50000 nM T99685 CVDG02 24905150 IC50 > 50000 nM T99685 CWH6C5 24905152 IC50 = 140 nM T99685 C0HE2Q 24905153 IC50 = 1700 nM T99685 C7QSC9 24905154 IC50 = 80 nM T99685 CO9D0K 24905155 IC50 = 100000 nM T99685 C5W9UR 24905157 IC50 = 934 nM T99685 CC1DA3 24905158 IC50 = 766 nM T99685 COW79F 24905159 IC50 = 5000 nM T99685 CFPA53 24905160 IC50 = 40000 nM T99685 C2O0JX 24905161 IC50 = 3800 nM T99685 CA72BE 24905162 IC50 = 4300 nM T99685 CQN6X9 24905163 IC50 = 4500 nM T99685 CD4O1F 24905165 IC50 = 100000 nM T99685 CKL48T 24905166 IC50 = 3500 nM T99685 C76VYL 24905167 IC50 = 12000 nM T99685 C7K5PU 24905168 IC50 = 4300 nM T99685 CZ57ID 24905169 IC50 = 8000 nM T99685 C2DHX9 24905170 IC50 = 5500 nM T99685 CSB96E 24905171 IC50 = 50000 nM T99685 CWZ0R2 24905172 IC50 = 1900 nM T99685 CY3B6M 24905175 IC50 = 8200 nM T99685 CW7UA3 24905176 IC50 = 404 nM T99685 CW1V0H 24905177 IC50 = 100000 nM T99685 CO6Y0L 24905178 IC50 = 5500 nM T99685 C60NQW 24905179 IC50 = 635 nM T99685 C4MO8B 24905180 IC50 = 192 nM T99685 COJI47 24905181 IC50 = 692 nM T99685 CS0B2C 24905182 IC50 = 10000 nM T99685 C1H4BT 24905183 IC50 = 1900 nM T99685 C4WHK9 24905184 IC50 = 10000 nM T99685 C7Q4MZ 24905185 IC50 = 300 nM T99685 CS4IP1 24905186 IC50 = 30000 nM T99685 C69QWO 24905187 IC50 = 576 nM T99685 C85ANB 24905188 IC50 = 364 nM T99685 CNHD75 24905189 IC50 = 2500 nM T99685 C9JUO2 24905190 IC50 = 8000 nM T99685 CPR03K 24905191 IC50 = 5400 nM T99685 CTAG19 24905193 IC50 = 407 nM T99685 C7VJM5 24905194 IC50 = 4500 nM T99685 CEP1L3 24905195 IC50 = 3400 nM T99685 CP68ZD 24905196 IC50 = 1600 nM T99685 C8Z0RJ 24905197 IC50 = 110 nM T99685 CN9RT0 24905198 IC50 = 18000 nM T99685 CHI78P 24905200 IC50 = 1900 nM T99685 CO6PE8 24905201 IC50 = 467 nM T99685 CZ63HS 24905202 IC50 = 60 nM T99685 C2X0FC 24905203 IC50 = 1200 nM T99685 C0WCE3 24905204 IC50 = 3000 nM T99685 CNK50B 24905205 IC50 = 550 nM T99685 C12DPB 24905206 IC50 = 596 nM T99685 C8N0RH 24905207 IC50 = 100000 nM T99685 CYA5G2 24905208 IC50 = 565 nM T99685 CDV2B4 24905209 IC50 = 8300 nM T99685 CEFK68 24905210 IC50 = 412 nM T99685 CUFP12 24905211 IC50 = 243 nM T99685 C0JG8L 24905212 IC50 = 493 nM T99685 CQ13ZI 24905215 IC50 = 2200 nM T99685 C6VI8F 24905216 IC50 = 113 nM T99685 CXNH25 24905217 IC50 = 1500 nM T99685 C2PN9S 24905218 IC50 = 632 nM T99685 C9O2AL 24905219 IC50 = 1100 nM T99685 CIT7U8 24905220 IC50 = 2200 nM T99685 CMD26S 24905221 IC50 = 457 nM T99685 C4R8WC 24905222 IC50 = 205 nM T99685 C47SHA 24905223 IC50 = 657 nM T99685 C1DY2R 24905224 IC50 = 1100 nM T99685 CS0XF9 24905225 IC50 = 6800 nM T99685 CG5VX2 24905226 IC50 = 8700 nM T99685 C57QEO 24905227 IC50 = 100000 nM T99685 C7CG5E 24905228 IC50 = 783 nM T99685 CHP5D1 24905229 IC50 = 1300 nM T99685 CXP09S 24905230 IC50 = 426 nM T99685 CY7XG1 24905231 IC50 = 3200 nM T99685 C7JFQ2 24905232 IC50 = 33 nM T99685 C2JM1P 24905233 IC50 = 10000 nM T99685 CC3BF0 24905234 IC50 = 100000 nM T99685 CE57FI 24905235 IC50 = 30000 nM T99685 CUP20O 24905236 IC50 = 100000 nM T99685 CLC6Q2 24905237 IC50 = 100000 nM T99685 C9M1GI 24905238 IC50 = 2400 nM T99685 CVD72F 24905239 IC50 = 1640 nM T99685 CK38IZ 24905240 IC50 = 596 nM T99685 CO2V5E 24905241 IC50 = 3600 nM T99685 CZBA19 24905244 IC50 = 7000 nM T99685 CQ8OI1 24905246 IC50 = 7600 nM T99685 CIF2J5 24905251 IC50 = 100000 nM T99685 CPTE58 24905252 IC50 = 3600 nM T99685 CP50RD 24905280 IC50 = 37 nM T99685 CG13ZM 24905281 IC50 = 911 nM T99685 CF0S6X 24905282 IC50 = 3300 nM T99685 C5HBL0 24905284 IC50 = 1200 nM T99685 C2Z5DN 24905285 IC50 = 4000 nM T99685 CL6GH8 24905286 IC50 = 710 nM T99685 CKYO98 24905287 IC50 = 33 nM T99685 CRNQ65 24905288 IC50 = 3 nM T99685 COD7I5 24905289 IC50 = 16 nM T99685 C4LP7E 24905290 IC50 = 861 nM T99685 CE9JC2 24905291 IC50 = 98 nM T99685 C2GI1R 24905292 IC50 = 100000 nM T99685 CHW8C4 24905293 IC50 = 20 nM T99685 CQF0H1 24905294 IC50 = 40 nM T99685 CNO7X0 24905295 IC50 = 130 nM T99685 C5WRG7 24905296 IC50 = 6500 nM T99685 CQ1S0U 24905297 IC50 = 4800 nM T99685 C4UES7 24905298 IC50 = 616 nM T99685 CMS69P 24905299 IC50 = 3200 nM T99685 CC0U5M 24905300 IC50 = 439 nM T99685 CW7X6S 24905301 IC50 = 100000 nM T99685 C97IQV 24905302 IC50 = 1800 nM T99685 CSJ47V 24905303 IC50 = 3000 nM T99685 CPN74C 24905304 IC50 = 15000 nM T99685 C5CS3N 24905305 IC50 = 4800 nM T99685 CK4XE9 24905307 IC50 = 50000 nM T99685 CTU6Z3 24905308 IC50 = 100000 nM T99685 C9SQX1 24905309 IC50 = 6500 nM T99685 CM75JP 24905310 IC50 = 5000 nM T99685 C9Q2BJ 24905311 IC50 = 3900 nM T99685 C9VUA1 24905312 IC50 = 2400 nM T99685 CU3RS1 24905313 IC50 = 5100 nM T99685 CYG3H2 24905314 IC50 = 30000 nM T99685 CV5Q7O 24905315 IC50 = 815 nM T99685 C8SA3O 24905316 IC50 = 170 nM T99685 CI5MN3 24905317 IC50 = 377 nM T99685 CJ1P7K 24905318 IC50 = 450 nM T99685 C1T6YQ 24905319 IC50 = 9200 nM T99685 CAU86X 24905320 IC50 = 1000 nM T99685 C54ISY 24905321 IC50 = 11000 nM T99685 C2GE5I 24905322 IC50 = 2000 nM T99685 C8D6YK 24905323 IC50 = 2900 nM T99685 C5NZH9 24905324 IC50 = 880 nM T99685 C9D6JR 24905325 IC50 = 1500 nM T99685 CLZT41 24905326 IC50 = 230 nM T99685 CW8FD3 24905327 IC50 = 1100 nM T99685 CHB7A2 24905328 IC50 = 2200 nM T99685 CA8EI3 24905329 IC50 = 833 nM T99685 CCQ0O7 24905330 IC50 = 100000 nM T99685 CJ81AS 24905331 IC50 = 548 nM T99685 C8PW4H 24905332 IC50 = 127 nM T99685 C2Y5TF 24905333 IC50 = 156 nM T99685 CH9FL5 24905334 IC50 = 1200 nM T99685 C1S0PC 24905335 IC50 = 1700 nM T99685 C8N9MV 24905336 IC50 = 1100 nM T99685 C9E8BJ 24905338 IC50 = 5000 nM T99685 CX85AC 24905341 IC50 = 5800 nM T99685 CKZ80E 24905342 IC50 = 14000 nM T99685 CO8SH1 24905343 IC50 = 3100 nM T99685 C7IZL6 24905344 IC50 = 5400 nM T99685 C3IYB2 24936050 IC50 = 0.08 nM T99685 CLD3X6 24936051 IC50 = 620 nM T99685 C98MEW 24946175 IC50 = 17 nM T99685 CC7H3U 24946706 IC50 = 880 nM T99685 CD5HQ0 24969301 IC50 > 10000 nM T99685 CCZO17 24970164 IC50 = 130 nM T99685 CXI65T 24983588 IC50 = 64 nM T99685 CH6Q7Y 24983749 IC50 = 176 nM T99685 C6Q8HD 24983903 IC50 = 273 nM T99685 C7NYZ4 24984057 IC50 = 231 nM T99685 CV79PK 24984058 IC50 = 21 nM T99685 CX24TD 24985362 IC50 = 60 nM T99685 CV5OB6 24985365 IC50 = 190 nM T99685 CBGM96 24985541 IC50 = 580 nM T99685 C2DLE6 24985542 IC50 > 10000 nM T99685 CORB97 24985709 IC50 = 1690 nM T99685 CQ39PB 24985717 IC50 = 5 nM T99685 C0G9DN 24985874 IC50 = 1360 nM T99685 CGSE92 25009673 Ki = 911 nM T99685 CB7VT5 25032306 Ki = 11.1 nM T99685 C2H3WJ 25032388 Ki = 2.54 nM T99685 C17PCM 25032389 Ki = 4.52 nM T99685 CM1GB6 25032390 Ki = 92.6 nM T99685 C0W2TF 25032391 Ki = 8.8 nM T99685 CCR6S7 25032392 Ki = 9.1 nM T99685 CBU2H9 25032644 Ki = 17 nM T99685 CHR51O 25057242 IC50 = 1800 nM T99685 C0T4NK 25070551 IC50 = 7200 nM T99685 C1UKQ4 25070552 IC50 = 2100 nM T99685 CZRA03 25070553 IC50 = 600 nM T99685 CO20FT 25070554 IC50 = 140 nM T99685 CL4B5Z 25070555 IC50 = 10500 nM T99685 C7U0SC 25070882 IC50 = 634 nM T99685 CCN36H 25071204 IC50 = 970 nM T99685 CQ7P4X 25071206 IC50 = 160 nM T99685 C14SFA 25071208 IC50 = 590 nM T99685 CNCJ40 25071516 IC50 = 570 nM T99685 CXWO13 25071518 IC50 = 310 nM T99685 CBH13R 25071519 IC50 = 160 nM T99685 CJM7O0 25071520 IC50 = 1700 nM T99685 C68PFD 25073081 IC50 = 170 nM T99685 CBJ20X 25073385 IC50 = 51 nM T99685 CZN7W0 25073388 IC50 = 152 nM T99685 C8DG4R 25109014 Ki = 59 nM T99685 CB3W1F 25109202 Ki = 42 nM T99685 CTO19H 25109378 Ki = 10 nM T99685 C83WVR 25109494 Ki = 30 nM T99685 CK2YI4 25168990 IC50 = 1.514 nM T99685 CC1D8V 25172062 IC50 = 300 nM T99685 CPW2D9 25172477 IC50 = 234 nM T99685 CXG59Q 25175568 IC50 = 303 nM T99685 C1C9ZF 25182020 IC50 = 913 nM T99685 CUA41N 25182022 IC50 > 6000 nM T99685 CX2N5M 25182023 IC50 > 6000 nM T99685 C46ZAW 25182142 IC50 > 6000 nM T99685 CP17FV 25182145 IC50 > 6000 nM T99685 CGQ56K 25182146 IC50 > 6000 nM T99685 C9G6DH 25182281 IC50 = 3010 nM T99685 CS07FL 25182282 IC50 > 6000 nM T99685 C2LYI1 25182285 IC50 > 6000 nM T99685 C7GAR5 25182286 IC50 > 6000 nM T99685 C9X3OT 25182424 IC50 > 6000 nM T99685 C0JBX1 25182427 IC50 > 6000 nM T99685 CAG4R1 25182562 IC50 > 6000 nM T99685 C5JD1M 25182565 IC50 > 6000 nM T99685 CWIH67 25182709 IC50 > 6000 nM T99685 C6O1VG 25182710 IC50 > 6000 nM T99685 C80UYN 25182711 IC50 > 6000 nM T99685 C8H9ET 25182714 IC50 > 6000 nM T99685 CD8M0G 25182867 IC50 > 6000 nM T99685 C9T6AZ 25182868 IC50 > 6000 nM T99685 C0S4YF 25182871 IC50 > 6000 nM T99685 CS4N6U 25183031 IC50 > 6000 nM T99685 CX8F3W 25183032 IC50 > 6000 nM T99685 C38MPQ 25195571 IC50 = 4.8 nM T99685 C1CL7V 25195572 IC50 = 2.4 nM T99685 CD4L2F 25195682 IC50 = 0.8 nM T99685 C4QTX9 25195788 IC50 = 0.3 nM T99685 CIRE40 25195789 IC50 = 23 nM T99685 CHJM38 25195893 IC50 = 65 nM T99685 C64SIJ 25195997 IC50 = 125 nM T99685 CB6CP3 25196219 IC50 = 16 nM T99685 CWN52I 25196221 IC50 = 1.4 nM T99685 C8RWY2 25196900 IC50 = 120 nM T99685 CNU28R 25197239 IC50 = 2.7 nM T99685 CMST49 25197240 IC50 = 0.8 nM T99685 CLW96O 25207689 Ki = 21 nM T99685 CRO09K 25211064 IC50 > 30000 nM T99685 C6MR3O 25229450 IC50 = 4.6 nM T99685 CQL23A 25229526 IC50 = 9 nM T99685 CWP29U 25242324 Ki = 30 nM T99685 C58WEU 25260757 IC50 = 0.21 nM T99685 C9V5KO 25260758 IC50 = 0.22 nM T99685 C8RYX7 25260759 IC50 = 0.24 nM T99685 C47RYE 25260913 IC50 = 0.19 nM T99685 C96OGS 25260915 IC50 = 0.38 nM T99685 CBCF51 25261227 IC50 = 0.5 nM T99685 C5DQF0 25261230 IC50 = 0.19 nM T99685 C4V2EJ 25261231 IC50 = 0.46 nM T99685 C3I9SN 25261388 IC50 = 0.23 nM T99685 C7SNP6 25261389 IC50 = 0.22 nM T99685 C4R3ZS 25261390 IC50 = 0.26 nM T99685 CUR93V 25261554 IC50 = 0.62 nM T99685 CCR83Z 25261555 IC50 = 0.11 nM T99685 C38UOX 25262174 IC50 = 0.48 nM T99685 CD27XK 25262616 IC50 = 0.74 nM T99685 CPLM23 25262617 IC50 = 0.6 nM T99685 CU6C8J 25262782 IC50 = 0.3 nM T99685 CT97DF 25262783 IC50 = 0.1 nM T99685 CFL6G2 25262946 IC50 = 1.34 nM T99685 CO4PL8 42606076 IC50 = 5100 nM T99685 C20VGT 42606077 IC50 = 10700 nM T99685 C7N5EC 42606078 IC50 = 10800 nM T99685 CI69YO 42606079 IC50 > 100000 nM T99685 C5L7IT 42606080 IC50 > 50000 nM T99685 CG04LZ 42606083 IC50 > 100000 nM T99685 C0WEU1 42606190 IC50 > 100000 nM T99685 CD6LN3 42606191 IC50 > 50000 nM T99685 CWR7P5 42606194 IC50 > 50000 nM T99685 CJ2GM1 42606195 IC50 > 50000 nM T99685 C61JUL 42606196 IC50 > 50000 nM T99685 C9GS8P 42606431 IC50 = 19100 nM T99685 CW63VM 42609338 Ki = 30 nM T99685 CYJK74 42632991 IC50 = 5900 nM T99685 CQW60S 42632992 IC50 = 3650 nM T99685 C2FIY7 42633175 IC50 = 2000 nM T99685 CL2XD7 42633904 IC50 > 4000 nM T99685 C9B0DZ 42633906 IC50 > 4000 nM T99685 CHP49D 42635321 IC50 = 355 nM T99685 C96ETP 42635322 IC50 = 1625 nM T99685 CZN3G1 42635323 IC50 = 5000 nM T99685 CCV0R1 42635502 IC50 = 430 nM T99685 CR8C3W 42635504 IC50 = 3600 nM T99685 C10RBA 42636535 IC50 > 5000 nM T99685 C3ROX1 44124863 IC50 = 0.4 nM T99685 C2YQX8 44125256 IC50 = 35 nM T99685 CV5O8L 44125375 IC50 = 20 nM T99685 C5JN4O 44125376 IC50 = 20 nM T99685 C0U2OY 44125377 IC50 = 6.6 nM T99685 C5CQK3 44138092 IC50 = 1 nM T99685 CP61GU 44156032 IC50 = 18 nM T99685 C3CBU7 44156033 IC50 = 500 nM T99685 C7XI2W 44156156 IC50 = 2 nM T99685 C63BLR 44156157 IC50 = 1 nM T99685 C19LGE 44158465 IC50 = 420 nM T99685 CG4DY5 44158569 IC50 = 95 nM T99685 CB46RQ 44159380 IC50 = 96 nM T99685 CIKM57 44180156 IC50 = 289 nM T99685 CXL61J 44181600 IC50 = 610 nM T99685 CO0YZ7 44182308 IC50 = 0.83 nM T99685 CS0M9A 44187604 IC50 = 0.63 nM T99685 C0BRI9 44187779 IC50 = 21 nM T99685 CDA81B 44187783 IC50 = 0.89 nM T99685 C0LB8S 44187784 IC50 = 3 nM T99685 CCTO21 44187951 IC50 = 2.55 nM T99685 CVYS60 44187952 IC50 = 0.5 nM T99685 C8X3UZ 44187955 IC50 = 2.2 nM T99685 CJU85Z 44188321 IC50 = 2.7 nM T99685 CHU02A 44188322 IC50 = 0.56 nM T99685 C69HQS 44188840 IC50 = 0.84 nM T99685 CD78AG 44188841 IC50 = 3.05 nM T99685 CY7EL1 44188842 IC50 = 0.51 nM T99685 C0SE1X 44188843 IC50 = 0.57 nM T99685 CG13ZF 44188844 IC50 = 0.32 nM T99685 CR0BF9 44189010 IC50 = 0.35 nM T99685 C71NFL 44189011 IC50 = 1.6 nM T99685 C39ABJ 44189192 IC50 = 0.31 nM T99685 CK73NR 44219749 IC50 = 4.3 nM T99685 C2V6WY 44232672 IC50 = 9.6 nM T99685 CA91IW 44232914 IC50 = 7 nM T99685 CN10TK 44232915 IC50 = 2450 nM T99685 CNY95J 44232916 IC50 = 46 nM T99685 COXT27 44232917 IC50 = 1.5 nM T99685 CFC2A1 44232918 IC50 = 1.4 nM T99685 CVN7P2 44233160 IC50 = 0.52 nM T99685 CQXD21 44233161 IC50 = 22 nM T99685 CI7N6F 44233162 IC50 = 2.1 nM T99685 CC6H5K 44233163 IC50 = 2 nM T99685 CSGQ48 44233164 IC50 = 1.1 nM T99685 CI65AN 44233388 IC50 = 1 nM T99685 CS9UA8 44233389 IC50 = 0.32 nM T99685 CZ3L7W 44233390 IC50 = 0.6 nM T99685 CA7R1U 44233391 IC50 = 0.5 nM T99685 CN4A7W 44233639 IC50 = 0.2 nM T99685 CWLA98 44233640 IC50 = 0.3 nM T99685 CXO1L7 44233641 IC50 = 0.34 nM T99685 CX7B1Y 44264159 IC50 < 10000 nM T99685 CVM4J9 44264177 IC50 < 10000 nM T99685 C8RNS0 44264540 IC50 < 10000 nM T99685 CA45LZ 44396556 IC50 = 1.45 nM T99685 C5EYH7 44396557 IC50 = 1.88 nM T99685 C52ZQN 44405685 IC50 = 5.8 nM T99685 C4QG5B 44405767 IC50 = 4.8 nM T99685 C2QF1N 44457157 IC50 = 829 nM T99685 C34HLQ 44457158 IC50 = 692 nM T99685 CSW53V 44457165 IC50 = 961 nM T99685 CZ4O2K 44457166 IC50 = 820 nM T99685 C6JS1G 44457167 IC50 = 890 nM T99685 CW5KH3 44457168 IC50 = 1870 nM T99685 CCBP46 44457169 IC50 > 1690 nM T99685 CWTU20 44457172 IC50 > 18700 nM T99685 C2QR9D 44457173 IC50 = 12600 nM T99685 C9H2FA 44457174 IC50 = 13900 nM T99685 C9X8CD 44457178 IC50 = 1210 nM T99685 CD4RP9 44457179 IC50 = 1350 nM T99685 C16ASL 44457183 IC50 = 3560 nM T99685 CA04RG 44457184 IC50 = 2330 nM T99685 C8INQ7 44457185 IC50 = 2290 nM T99685 C0UBI8 44457188 IC50 = 767 nM T99685 CGCS67 44457189 IC50 = 1480 nM T99685 C9WG2B 44457191 IC50 = 3570 nM T99685 C4OK8P 44457192 IC50 = 878 nM T99685 CHSE37 44457195 IC50 = 1470 nM T99685 CN9H7F 44457201 IC50 = 1800 nM T99685 CI6G5C 44457211 IC50 = 960 nM T99685 C9N4PA 44457212 IC50 = 831 nM T99685 CB70NU 44457213 IC50 = 816 nM T99685 CY4H8C 44457218 IC50 = 568 nM T99685 C0RN9S 44457220 IC50 = 822 nM T99685 C2JV8Y 44457231 IC50 = 2450 nM T99685 CQD4T3 44457232 IC50 = 1690 nM T99685 CT02VO 44457235 IC50 = 249 nM T99685 CB2J6E 44457236 IC50 = 619 nM T99685 CG7YT9 44457237 IC50 = 1200 nM T99685 CVG75D 44473371 IC50 = 0.5 nM T99685 CX3FK1 44513884 IC50 = 1.2 nM T99685 CL4RO5 44513885 IC50 = 1.2 nM T99685 C6RC9J 44513886 IC50 = 3.9 nM T99685 CGS7Q4 44513887 IC50 = 1.7 nM T99685 CSVD32 44513888 IC50 = 6.3 nM T99685 CLN2M5 44514201 IC50 = 3.9 nM T99685 C2Y8ML 44514203 IC50 = 6.7 nM T99685 CA9H8D 44514205 IC50 = 9.3 nM T99685 C01ZJI 44514208 IC50 = 0.3 nM T99685 CZ8WK6 44514210 IC50 = 0.4 nM T99685 CI8H3K 44514481 IC50 = 10 nM T99685 C51SEJ 44515083 IC50 = 1.8 nM T99685 CXBV98 44515084 IC50 = 1.9 nM T99685 C73HNB 44515696 IC50 = 2.5 nM T99685 CB7XW5 44516307 IC50 = 1.5 nM T99685 C4W5EM 44516309 IC50 = 1.4 nM T99685 C8VAU1 44516310 IC50 = 0.7 nM T99685 C8I1ZB 44516311 IC50 = 0.6 nM T99685 CSJ95V 44516635 IC50 = 0.8 nM T99685 CV6Z0N 44516636 IC50 = 0.7 nM T99685 CB3MV8 44517288 IC50 = 1.3 nM T99685 CDEQ97 44520808 IC50 = 215 nM T99685 CT7DW6 44520809 IC50 = 49 nM T99685 C3T2YD 44520810 IC50 = 4 nM T99685 CJP71L 44520811 IC50 = 6 nM T99685 CB4RN0 44520812 IC50 = 83 nM T99685 CGQ1F8 44520814 IC50 = 695 nM T99685 C2W5QS 44520815 IC50 = 7300 nM T99685 CN78XU 44520816 IC50 = 5950 nM T99685 C1TI9F 44520817 IC50 = 190 nM T99685 CHS6C1 44520818 IC50 = 130 nM T99685 CKP60Q 44520819 IC50 = 145 nM T99685 C0XEA9 44520820 IC50 = 88 nM T99685 CFE63J 44520821 IC50 = 230 nM T99685 CV43BN 44520822 IC50 = 380 nM T99685 CYU2B5 44520824 IC50 = 170 nM T99685 C73ZYA 44520825 IC50 = 4 nM T99685 CB25DI 44539683 IC50 = 1.4 nM T99685 CNWO35 44539684 IC50 = 0.67 nM T99685 C8MTO3 44539685 IC50 = 7.5 nM T99685 CTQ06N 44539783 IC50 = 42 nM T99685 C3D8CF 44540543 IC50 = 0.46 nM T99685 C0Z3QI 44540642 IC50 = 37 nM T99685 C3Z7GL 44540644 IC50 = 0.94 nM T99685 CGB2A8 44540925 IC50 = 9.5 nM T99685 CFI4O2 44541101 IC50 = 11 nM T99685 CW19QS 44544943 Ki = 950 nM T99685 C6L4SV 44545041 Ki = 72 nM T99685 C0IX1C 44545849 IC50 = 3 nM T99685 C6HC3L 44548482 IC50 = 5.3 nM T99685 CH3L9P 44551660 IC50 = 4590 nM T99685 CYMD49 44552663 IC50 = 1650 nM T99685 C6B7LH 44552664 IC50 = 11 nM T99685 C3QZX0 44552666 IC50 = 18 nM T99685 C64OQC 44552667 IC50 = 9 nM T99685 C7LG6Q 44552844 IC50 = 118 nM T99685 C9T2CZ 44552845 IC50 = 18 nM T99685 CXLD75 44552846 IC50 = 108 nM T99685 CALT95 44554240 IC50 = 130 nM T99685 CVDA08 44554755 IC50 = 190 nM T99685 C25EGX 44554909 IC50 = 280 nM T99685 C6VR1P 44554910 IC50 = 123 nM T99685 CR4J0X 44554913 IC50 = 3700 nM T99685 CWV2T9 44554915 IC50 = 153 nM T99685 CCW12H 44555222 IC50 = 265 nM T99685 CTM8S9 44555225 IC50 = 2125 nM T99685 C7PSO6 44555226 IC50 = 430 nM T99685 C3VRO9 44557921 IC50 > 10000 nM T99685 C8A5RT 44577639 IC50 > 15000 nM T99685 C5VNA7 44599029 IC50 = 2 nM T99685 CCFX21 44599203 IC50 = 1 nM T99685 CU5YK1 44599206 IC50 = 1.7 nM T99685 C4OP3Y 44599690 IC50 = 0.6 nM T99685 C7H0XM 44599855 IC50 = 1.7 nM T99685 CL73YV 44600010 IC50 = 0.5 nM T99685 C54ZQB 44600166 IC50 = 0.9 nM T99685 C2ZYD0 44600649 IC50 = 0.4 nM T99685 C3R2PX 44600650 IC50 = 205 nM T99685 C8AT9I 44600651 IC50 = 64 nM T99685 C5JL6C 44600806 IC50 = 1 nM T99685 CJUQ51 44600808 IC50 > 800 nM T99685 C0BXS4 44600809 IC50 > 800 nM T99685 CA9LP4 44600952 IC50 = 3 nM T99685 CFK83C 44600954 IC50 = 7 nM T99685 CX30VY 44600955 IC50 = 2 nM T99685 C9N1SY 44600956 IC50 = 8 nM T99685 CUI9Y8 44601112 IC50 = 30 nM T99685 CBV38N 44601113 IC50 = 33 nM T99685 CA3K8E 44601278 IC50 = 7 nM T99685 CZX94G 44601279 IC50 = 52 nM T99685 CD1A2Z 44601448 IC50 = 11 nM T99685 CB12CS 44601449 IC50 = 24 nM T99685 CIDT64 44601450 IC50 = 14 nM T99685 CWY15L 44604823 IC50 = 2.6 nM T99685 CN9ZD0 44604824 IC50 = 0.7 nM T99685 CL3S1F 44604825 IC50 = 23 nM T99685 C28QLM 44605035 IC50 = 4.6 nM T99685 C75XHS 44605037 IC50 = 0.4 nM T99685 CFN95D 44605038 IC50 = 0.3 nM T99685 CD8Q9Z 44605039 IC50 = 0.1 nM T99685 CI70YP 44605246 IC50 = 0.7 nM T99685 C36ZFK 44605247 IC50 = 0.8 nM T99685 CEK25C 44605248 IC50 = 0.6 nM T99685 C3F4UX 44605249 IC50 = 0.2 nM T99685 CQ0FZ7 44605426 IC50 = 0.3 nM T99685 CC7G2L 44605427 IC50 = 0.5 nM T99685 CDLP04 44605428 IC50 = 0.7 nM T99685 CSKN09 44605429 IC50 = 0.5 nM T99685 CA79QG 44605430 IC50 = 0.6 nM T99685 CM49FO 44605789 IC50 = 2.3 nM T99685 C3DK5F 44605790 IC50 = 1.9 nM T99685 C9Z4TY 44605791 IC50 = 0.62 nM T99685 C9F8JY 44605792 IC50 = 0.87 nM T99685 CGT58A 44606131 IC50 = 0.6 nM T99685 CTO96K 44606133 IC50 = 0.23 nM T99685 CH7O9Y 44606302 IC50 = 1.2 nM T99685 C8Y4FE 44606303 IC50 = 0.58 nM T99685 C4PEO6 44606304 IC50 = 1 nM T99685 CG04KF 44606474 IC50 = 5.5 nM T99685 C86RYX 44606475 IC50 = 91 nM T99685 CNI9G3 44606476 IC50 = 1.9 nM T99685 CE90UX 44606477 IC50 = 53 nM T99685 CQIY50 44606640 IC50 = 17 nM T99685 C1ML5R 44606641 IC50 = 1.8 nM T99685 C35QOE 44606642 IC50 = 1.8 nM T99685 CWQ67K 44606643 IC50 = 1.2 nM T99685 CY0QH9 44606644 IC50 = 0.28 nM T99685 CFQT17 44606818 IC50 = 480 nM T99685 C84TLP 44606820 IC50 = 170 nM T99685 C3H4EB 44606823 IC50 = 27 nM T99685 CD4A8G 44606998 IC50 = 111 nM T99685 C80RQK 44606999 IC50 = 73 nM T99685 CFW9G3 44607000 IC50 = 9.6 nM T99685 CHL59X 44607001 IC50 = 113 nM T99685 C7H3RM 44607002 IC50 = 145 nM T99685 C2TJ3K 44607003 IC50 = 16 nM T99685 CHM5T4 44607180 IC50 = 20 nM T99685 C85XWN 44607181 IC50 = 200 nM T99685 C52ILQ 44607183 IC50 = 12 nM T99685 C2UP6C 44607528 IC50 = 76 nM T99685 CH6OY3 44607529 IC50 = 84 nM T99685 CH6V9F 44608754 IC50 = 3.9 nM T99685 C0IY9N 44608757 IC50 = 5.3 nM T99685 C90ITS 44608915 IC50 = 3.9 nM T99685 CZH1P9 44609387 IC50 = 5 nM T99685 CNDX48 44609388 IC50 = 37 nM T99685 C4TS8G 44610775 IC50 = 21 nM T99685 CAE82W 44623107 IC50 < 1 nM T99685 CYGA93 44814560 Ki = 12 nM T99685 CV24XP 44814563 Ki = 6.6 nM T99685 C37AQP 44815590 Ki = 9.6 nM T99685 CQVB69 44816122 Ki = 17 nM T99685 CT2Y5W 44816299 Ki = 122 nM T99685 C27ZIX 44816464 Ki = 5.1 nM T99685 C6GA8J 44816634 Ki = 1500 nM T99685 CIS31K 44817154 Ki = 21 nM T99685 C54IUP 44818842 IC50 = 250 nM T99685 C16IMZ 44819024 IC50 = 2.95 nM T99685 CN38JF 44819199 IC50 = 0.57 nM T99685 CVW6L8 44819200 IC50 = 3.7 nM T99685 CZ7M6D 44819201 IC50 = 0.39 nM T99685 C7MU8J 44819203 IC50 = 0.75 nM T99685 C8FU0W 44819375 IC50 = 1.21 nM T99685 C4N8CK 44819376 IC50 = 1.1 nM T99685 C0U1IR 45139233 Ki = 500 nM T99685 CK49WN 45139234 Ki = 3900 nM T99685 CYP0M7 45254032 IC50 = 5.4 nM T99685 C1BRW8 45254590 Ki = 4.51 nM T99685 CQ92ME 45379087 Ki = 396 nM T99685 C5I1VH 45379222 IC50 = 11.3 nM T99685 CA4JZ8 45379223 IC50 = 2.3 nM T99685 C12QFV 45480167 Ki = 840 nM T99685 C4V5DT 45482916 IC50 = 0.62 nM T99685 CAL96M 45482923 IC50 = 0.16 nM T99685 C8T6ML 45482926 IC50 = 0.22 nM T99685 C5C2YW 45482931 IC50 = 84 nM T99685 CP45HK 45482935 IC50 = 0.17 nM T99685 CR93VD 45482947 IC50 = 0.2 nM T99685 CDXB49 45482952 IC50 = 0.56 nM T99685 CCS97L 45482982 IC50 = 0.2 nM T99685 CX4TC8 45483330 IC50 = 575 nM T99685 C28OEC 45487702 IC50 = 1500 nM T99685 C38HVQ 45487703 IC50 = 5500 nM T99685 COXA34 45487715 IC50 = 510 nM T99685 C36DZY 45487716 IC50 = 520 nM T99685 CJ7U6H 45487737 IC50 > 10000 nM T99685 CNHR02 45487749 IC50 = 570 nM T99685 CV81ML 45487755 IC50 = 180 nM T99685 CF3TV5 45488020 IC50 = 13 nM T99685 CPLM59 45488021 IC50 = 51 nM T99685 CIL9W1 45488031 IC50 = 1.1 nM T99685 C2Q9ID 45488032 IC50 = 0.2 nM T99685 CA98FY 45488033 IC50 = 0.7 nM T99685 CH07NQ 45488034 IC50 = 0.8 nM T99685 CB8DE0 45488052 IC50 = 0.1 nM T99685 CF3LV9 45488056 IC50 = 2.7 nM T99685 CCL46I 45488057 IC50 = 0.7 nM T99685 CP58QK 45488058 IC50 = 0.1 nM T99685 C9S4MU 45488059 IC50 = 0.3 nM T99685 C0V7UL 45488060 IC50 = 0.2 nM T99685 C8YEC5 45488061 IC50 = 0.2 nM T99685 C6RTH4 45488066 IC50 = 0.9 nM T99685 CWN8V6 45488069 IC50 = 1.5 nM T99685 C1YM6P 45488070 IC50 = 0.3 nM T99685 CNK52A 45488071 IC50 = 1 nM T99685 CO8T6V 45488077 IC50 = 0.3 nM T99685 CBAT68 45488078 IC50 = 6 nM T99685 CZ68MG 45488079 IC50 = 0.6 nM T99685 CFOH35 45488080 IC50 = 0.2 nM T99685 CE3Q7D 45488081 IC50 = 1.7 nM T99685 CI3FZ2 45488082 IC50 = 0.9 nM T99685 CV1U7I 46180604 Ki = 29 nM T99685 CZGB46 46180666 IC50 = 750 nM T99685 CASO36 46182743 Ki = 6.8 nM T99685 C4HFV9 46190734 IC50 = 1.8 nM T99685 CTZD58 46190735 IC50 = 1.1 nM T99685 C61ZLI 46190736 IC50 > 4000 nM T99685 C0V5FS 46190794 IC50 = 66 nM T99685 CA36SV 46191509 IC50 = 336 nM T99685 C5V1DM 46191571 IC50 = 287 nM T99685 CV89YR 46191573 IC50 = 396 nM T99685 C2VJQ1 46191628 IC50 = 230 nM T99685 CR9SZ1 46191757 IC50 = 66.5 nM T99685 CP8DY9 46191758 IC50 = 45.9 nM T99685 C6H3GT 46196486 IC50 = 0.8 nM T99685 CL08DK 46201895 IC50 = 1.4 nM T99685 CL4U2V 46202650 Ki = 110 nM T99685 CX3D9U 46202651 Ki = 106 nM T99685 C9PC6U 46202652 Ki = 203 nM T99685 CHDX80 46202976 IC50 = 729 nM T99685 CI47RP 46206016 IC50 = 23 nM T99685 C3Z6BX 46206784 IC50 = 1 nM T99685 C1D4TK 46214389 IC50 = 90 nM T99685 C1RNM6 46214392 IC50 = 122 nM T99685 C93ZNA 46215208 IC50 = 68 nM T99685 CX8S2G 46215210 IC50 = 18 nM T99685 CF57GK 46215462 IC50 > 10000 nM T99685 CGMS50 46215563 IC50 = 90 nM T99685 CRBF57 46215564 IC50 = 108 nM T99685 CO1D6B 46215565 IC50 = 149 nM T99685 CDA3R9 46220225 Ki > 10000 nM T99685 CIJ5V9 46224766 IC50 = 720 nM T99685 CIPV59 46224808 IC50 = 2050 nM T99685 C4SQY2 46225156 IC50 = 3.3 nM T99685 CL89JZ 46225157 IC50 = 2.5 nM T99685 CFB7Y4 46225158 IC50 = 7.2 nM T99685 C65IPQ 46225280 IC50 = 870 nM T99685 C8A7QJ 46225281 IC50 = 200 nM T99685 CPL45H 46225307 IC50 = 8900 nM T99685 CU12LG 46227561 IC50 = 35 nM T99685 CU0T1P 46227563 IC50 = 100 nM T99685 CK20PN 46227564 IC50 = 22 nM T99685 C3VB6I 46227571 IC50 = 26.5 nM T99685 CS03RK 46227572 IC50 = 0.29 nM T99685 CO4J6R 46227578 IC50 = 11 nM T99685 CO14HC 46227579 IC50 = 0.44 nM T99685 CM1A2S 46227582 IC50 = 20 nM T99685 CT2CH5 46227596 IC50 = 0.9 nM T99685 CG26LH 46227597 IC50 = 1.4 nM T99685 CXW1N8 46227599 IC50 = 0.7 nM T99685 CO64ZL 46227600 IC50 = 0.7 nM T99685 CBF0O4 46227603 IC50 = 16 nM T99685 C2Z4WI 46227604 IC50 = 1 nM T99685 C76PKV 46227605 IC50 = 4.7 nM T99685 C3JK1T 46227606 IC50 = 0.6 nM T99685 CV9O8I 46227607 IC50 = 3.7 nM T99685 CW25EH 46227608 IC50 = 0.45 nM T99685 C5FU9E 46227614 IC50 = 58 nM T99685 C59UJH 46227615 IC50 = 0.34 nM T99685 CS3A9G 46227620 IC50 = 0.68 nM T99685 CG29EB 46227625 IC50 = 1.25 nM T99685 CI9CJ1 46227632 IC50 = 57 nM T99685 CL34IK 46227801 IC50 = 290 nM T99685 C6D2RL 46227820 IC50 = 90 nM T99685 CSIK15 46228569 IC50 = 460 nM T99685 C18WPC 46232643 IC50 = 0.12 nM T99685 CF4WB3 46232644 IC50 = 2.85 nM T99685 C7LKA5 46232645 IC50 = 14.5 nM T99685 C3ZP0G 46232682 IC50 = 0.33 nM T99685 CLE2O9 46232721 IC50 = 0.74 nM T99685 C4IA5M 46232759 IC50 = 1.19 nM T99685 C64HAE 46232760 IC50 = 0.26 nM T99685 CIMH64 46232761 IC50 = 0.22 nM T99685 C47ZSV 46232801 IC50 = 0.22 nM T99685 CVF7G6 46232802 IC50 = 0.16 nM T99685 CXP84Y 46232803 IC50 = 0.12 nM T99685 CT2O8D 46232804 IC50 = 0.12 nM T99685 CL7C2K 46244173 IC50 = 180 nM T99685 C2NH0A 46244259 IC50 = 230 nM T99685 CVJM38 46244260 IC50 = 3300 nM T99685 C79JGP 46830152 IC50 = 5.4 nM T99685 CC62SY 46830153 IC50 = 9 nM T99685 CU4T7F 46830277 IC50 = 3.1 nM T99685 CZ3WS1 46861592 IC50 = 0.2 nM T99685 C7H4YM 46865419 IC50 > 10000 nM T99685 CRO8W0 46865423 IC50 = 3 nM T99685 C47VTS 46865424 IC50 = 10 nM T99685 C7Q4OP 46865531 Ki = 5 nM T99685 C7T4RN 46865885 IC50 = 1 nM T99685 CO3P0J 46866604 IC50 = 0.46 nM T99685 CQ2Y1V 46866705 Ki = 1.42 nM T99685 C62NFQ 46883920 IC50 = 5.6 nM T99685 CKJ2D4 46883989 IC50 = 57 nM T99685 C82RWD 46883990 IC50 = 3500 nM T99685 CE3B7R 46883991 IC50 = 3.45 nM T99685 CP9JO4 46884017 IC50 = 145 nM T99685 C18KOY 46884018 IC50 = 14.3 nM T99685 C9RD8J 46884019 IC50 = 29 nM T99685 CP3C4Z 46884064 IC50 = 71 nM T99685 C65AQI 46884065 IC50 = 10.5 nM T99685 C7NK1H 46884066 IC50 = 115 nM T99685 C3BV5E 46884067 IC50 = 18 nM T99685 C9LB7I 46884068 IC50 = 17 nM T99685 CLOR10 46884069 IC50 = 70 nM T99685 CE70MJ 46884070 IC50 = 8.2 nM T99685 CIAK59 46884071 IC50 = 47.5 nM T99685 CO09QJ 46884072 IC50 = 8.2 nM T99685 CK95YV 46884073 IC50 = 10.9 nM T99685 CUI09D 46884074 IC50 = 9.3 nM T99685 CUL4I2 46884075 IC50 = 8.4 nM T99685 C9MHF4 46884076 IC50 = 102.5 nM T99685 CHM48L 46884077 IC50 = 13 nM T99685 C6MZ1J 46884121 IC50 = 800 nM T99685 C96FTP 46884122 IC50 = 33 nM T99685 C5RM6X 46884123 IC50 = 42 nM T99685 CKT35D 46884156 IC50 = 19 nM T99685 CFP9B5 46884157 IC50 = 0.55 nM T99685 CI3U2Q 46884158 IC50 = 0.5 nM T99685 CTVN70 46884203 IC50 = 0.56 nM T99685 C4FC9H 46884204 IC50 = 2 nM T99685 CEJ9C3 46884242 IC50 = 1 nM T99685 C8S5TR 46884243 IC50 = 0.39 nM T99685 CU93BN 46884282 IC50 = 1.85 nM T99685 C2H5CE 46884283 IC50 = 4.55 nM T99685 CWFH78 46884284 IC50 = 18 nM T99685 CZ5M8O 46884285 IC50 = 180 nM T99685 CV3C0K 46884353 IC50 = 0.72 nM T99685 CZV8T9 46884354 IC50 = 17 nM T99685 CO9W8A 46884355 IC50 = 19 nM T99685 CLA01F 46884356 IC50 = 2.2 nM T99685 CO1D2H 46884404 IC50 = 0.38 nM T99685 CB6YM8 46884405 IC50 = 2.1 nM T99685 CL8PR5 46884406 IC50 = 2.75 nM T99685 CY9M0N 46884525 IC50 = 0.18 nM T99685 CH0QN3 46884526 IC50 = 0.7 nM T99685 CAU6E8 46884527 IC50 = 5.4 nM T99685 CA2U0D 46884528 IC50 = 6.6 nM T99685 C5JBC1 46884529 IC50 = 8.8 nM T99685 CH2RD9 46884530 IC50 = 1.2 nM T99685 CWHK39 46884531 IC50 = 0.7 nM T99685 CSQ5I3 46884532 IC50 = 0.52 nM T99685 CS0Q3T 46884533 IC50 = 0.535 nM T99685 CO5H2J 46884534 IC50 = 0.56 nM T99685 C31KXQ 46884535 IC50 = 0.88 nM T99685 C86PXB 46884536 IC50 = 0.56 nM T99685 C6TI7E 46884537 IC50 = 0.81 nM T99685 CRW39C 46884538 IC50 = 0.34 nM T99685 C02IJK 46884539 IC50 = 0.14 nM T99685 C4SX6O 46884540 IC50 = 0.7 nM T99685 CE5S7W 46884541 IC50 = 0.4 nM T99685 CAS1R6 46884542 IC50 = 1.2 nM T99685 C87UVQ 46884543 IC50 = 1.25 nM T99685 C2RJ4E 46884544 IC50 = 0.9 nM T99685 CE8YC5 46884545 IC50 = 0.42 nM T99685 CM3C9U 46884546 IC50 = 0.1 nM T99685 CGY1E3 46884547 IC50 = 1.7 nM T99685 CUPR76 46885272 IC50 = 0.25 nM T99685 CHP18Q 46885273 IC50 = 0.57 nM T99685 CY89OZ 46885274 IC50 = 0.57 nM T99685 CZ1XR9 46885275 IC50 = 1 nM T99685 C9N5RS 46885276 IC50 = 1.1 nM T99685 CZYO07 46885277 IC50 = 0.89 nM T99685 C1Y7QN 46885278 IC50 = 1.6 nM T99685 CNLX49 46885279 IC50 = 0.9 nM T99685 CSA92E 46885280 IC50 = 0.8 nM T99685 CL4ZI9 46885281 IC50 = 0.26 nM T99685 CN3RH4 46885425 IC50 = 9200 nM T99685 CLA40T 46885426 IC50 = 11000 nM T99685 COL95X 46885494 IC50 = 5000 nM T99685 CVWU94 46885495 IC50 = 500 nM T99685 CC8T1E 46885496 IC50 = 190 nM T99685 CM8JX9 46885534 IC50 = 22 nM T99685 CCS20H 46885565 IC50 = 1 nM T99685 CG47YP 46885566 IC50 = 62 nM T99685 C4R3XP 46885599 IC50 = 4 nM T99685 C3SMV1 46885600 IC50 = 96 nM T99685 CV5MK6 46885601 IC50 = 215 nM T99685 C2M1DN 46885624 IC50 = 108 nM T99685 C42WVO 46885648 IC50 = 7 nM T99685 C0ZV8M 46886360 Ki = 10 nM T99685 C1JS5T 46886361 Ki = 50 nM T99685 CGRO36 46886375 Ki = 4 nM T99685 CZR3V2 46886410 Ki = 4 nM T99685 C4PRU3 46891423 IC50 = 1.3 nM T99685 CXPZ24 46891467 IC50 = 5.2 nM T99685 C9G4IW 46891468 IC50 = 2.4 nM T99685 C4IW0N 46891469 IC50 = 1.5 nM T99685 CF17MQ 46891470 IC50 = 4.2 nM T99685 CRHK80 46891471 IC50 = 3.8 nM T99685 C9SUH8 46891472 IC50 = 1.1 nM T99685 CGME41 46891473 IC50 = 2.5 nM T99685 C3HMQ2 46891474 IC50 = 0.3 nM T99685 CARY94 46891475 IC50 > 4000 nM T99685 CP38DV 46891889 Ki = 9 nM T99685 CB6Z8P 46892208 IC50 = 1300 nM T99685 CZX46Y 46892342 IC50 = 1500 nM T99685 C5FN6I 46892845 IC50 = 390 nM T99685 CQ32BN 46892970 IC50 = 150 nM T99685 COJA32 46892971 IC50 = 8 nM T99685 C5QFB3 46893088 IC50 = 27 nM T99685 C1Q8HJ 46893484 IC50 = 370 nM T99685 CO5ZE0 46893618 IC50 = 43 nM T99685 CS30AI 46893754 IC50 = 31 nM T99685 C8ESU7 46912801 Ki = 10 nM T99685 C3HG6N 46913071 Ki = 140 nM T99685 CDGN94 46913265 Ki = 12 nM T99685 CIM9S2 46913471 Ki = 12 nM T99685 CPO1N7 46927938 Ki = 4880 nM T99685 CFO9X3 46946049 IC50 = 989 nM T99685 CL84AF 46946248 IC50 > 10000 nM T99685 CF14PE 46947264 IC50 = 0.42 nM T99685 CMRT49 49780177 IC50 = 966 nM T99685 C2Y9OC 49780178 IC50 = 3810 nM T99685 C4T2GU 49780179 IC50 = 13.5 nM T99685 CLW50G 49780380 IC50 = 78.9 nM T99685 CP92MJ 49780381 IC50 = 93.8 nM T99685 C1TIH2 49780382 IC50 = 3440 nM T99685 C64MFW 49780383 IC50 = 33.2 nM T99685 CL1W9U 49780384 IC50 = 662 nM T99685 CV0I7K 49780592 IC50 = 213 nM T99685 CZ2T5F 49780593 IC50 = 82.6 nM T99685 CKMO53 49780594 IC50 = 214 nM T99685 C3WAJ9 49780595 IC50 = 25.8 nM T99685 CQB86T 49780596 IC50 = 239 nM T99685 CA1IQ0 49780810 IC50 = 95 nM T99685 C0N6SF 49780811 IC50 = 6.84 nM T99685 C5RBK7 49780812 IC50 = 3.6 nM T99685 CG82WE 49780813 IC50 = 0.57 nM T99685 C7AY6O 49781041 IC50 = 389 nM T99685 C91BTF 49781042 IC50 = 1.26 nM T99685 C6QV0A 49781043 IC50 = 21.4 nM T99685 CGU7Y0 49781044 IC50 = 4.25 nM T99685 C74ZTC 49781256 IC50 = 26.6 nM T99685 CC05VI 49781257 IC50 = 51.9 nM T99685 CHX76J 49784892 IC50 = 7800 nM T99685 CA1H8S 49784893 IC50 > 10000 nM T99685 CP2QD0 49784894 IC50 = 4800 nM T99685 CTZG05 49784988 IC50 = 7200 nM T99685 CE9AC5 49785078 IC50 = 560 nM T99685 CG2IO7 49785079 IC50 = 530 nM T99685 C8EYN4 49785083 IC50 > 10000 nM T99685 CBNZ47 49785166 IC50 > 10000 nM T99685 CZI34V 49785167 IC50 > 10000 nM T99685 CJK65T 49785253 IC50 = 360 nM T99685 CXK8F5 49785436 IC50 > 10000 nM T99685 CWL5C6 49785518 IC50 > 10000 nM T99685 C3NV0J 49785827 IC50 = 200 nM T99685 C0OZM2 49785828 IC50 > 10000 nM T99685 C1AR4G 49785829 IC50 > 10000 nM T99685 C39HAK 49785832 IC50 > 10000 nM T99685 CA53NO 49788443 IC50 = 237 nM T99685 C9K1XO 49800133 Ki = 0.85 nM T99685 C3D2RG 49800134 Ki = 5.11 nM T99685 CQ93PT 49800135 Ki = 5 nM T99685 CWI3E0 49800136 Ki = 0.8 nM T99685 C9ZW3R 49835055 IC50 = 12 nM T99685 CI6B7G 49835106 IC50 = 37 nM T99685 CN2E0P 49835107 IC50 = 13 nM T99685 CV50DY 49835108 IC50 = 198 nM T99685 CTM6U1 49835172 IC50 = 121 nM T99685 CL6V8Y 49835227 IC50 = 35 nM T99685 C90XTJ 49835286 IC50 = 3 nM T99685 CA4NH7 49850583 IC50 = 5000 nM T99685 CT4Y6E 49852123 IC50 > 50000 nM T99685 CXOH76 49855456 Ki = 3.2 nM T99685 C08PSJ 49855457 Ki = 3.6 nM T99685 CFHP43 49855648 Ki = 1.7 nM T99685 CEPR84 49856040 Ki = 1.3 nM T99685 CP2LC8 49857180 Ki = 10 nM T99685 CWT1P9 49857571 Ki = 1.4 nM T99685 CJ21VU 49857572 Ki = 4.4 nM T99685 C5E0JI 49858150 Ki = 0.7 nM T99685 C6JBA1 49858345 Ki = 3 nM T99685 C1C2UI 49858346 Ki = 1.6 nM T99685 CY8MP7 49867926 IC50 = 190 nM T99685 C25YNT 50940492 Ki = 5 nM T99685 C2Q0GE 50990922 IC50 = 93 nM T99685 CKY3V1 50990924 IC50 = 2 nM T99685 CGQ49I 51003483 Ki = 3 nM T99685 C0HWJ7 51003484 Ki = 13 nM T99685 CHP3Z4 51003485 Ki = 265 nM T99685 CPA8N1 51039139 Ki = 8 nM T99685 CLZ8N6 51352027 IC50 = 6.31 nM T99685 C73ANH 51353707 IC50 = 57 nM T99685 CI4A6R 51353708 IC50 = 285 nM T99685 CJ4ZL6 51353709 IC50 = 262 nM T99685 CDLF71 51353710 IC50 = 45 nM T99685 C04EVK 51353711 IC50 > 6000 nM T99685 CD6AL8 51353712 IC50 = 47 nM T99685 CPQ1G6 51354021 IC50 = 719 nM T99685 CVK95R 51354022 IC50 = 65 nM T99685 CHKA96 51354023 IC50 = 269 nM T99685 CRL1B8 51354025 IC50 > 6000 nM T99685 C6VD0B 51354313 IC50 = 29 nM T99685 CJC90Y 51354315 IC50 = 11 nM T99685 COH9L7 51354317 IC50 = 15 nM T99685 CV6I5D 51354595 IC50 = 1500 nM T99685 C1V6RN 51354597 IC50 = 1.6 nM T99685 CZ32XV 51354599 IC50 = 6 nM T99685 C8WEN4 51354600 IC50 = 2.1 nM T99685 C76KOV 51354878 IC50 < 1 nM T99685 CA3O2L 51354879 IC50 < 1 nM T99685 C0O2PW 51354880 IC50 = 1.6 nM T99685 C3JV4L 51354881 IC50 < 1 nM T99685 C6NL1Z 51354882 IC50 < 1 nM T99685 CPWD73 51354883 IC50 < 1 nM T99685 C9CYA1 51355056 Ki = 150 nM T99685 C6E9WP 51355057 Ki = 30 nM T99685 C4QE1V 51355058 Ki = 69 nM T99685 CB10AP 51355171 IC50 = 2.1 nM T99685 CKE42Q 51355172 IC50 = 2.1 nM T99685 CZF89J 51355173 IC50 = 1.1 nM T99685 CQF0J9 51355174 IC50 = 2.3 nM T99685 CO7M9F 51355343 Ki = 4 nM T99685 CJ0KM6 51355344 Ki = 120 nM T99685 CT0V8F 51355345 Ki = 40 nM T99685 C0R8XN 51355348 Ki = 2 nM T99685 C7KT4Z 51355620 Ki = 1 nM T99685 CI71WE 51355621 Ki = 28 nM T99685 CLH35Z 51355622 Ki = 30 nM T99685 C2ODW5 51357942 IC50 > 6000 nM T99685 CSR12N 51357943 IC50 > 6000 nM T99685 CT8LF4 51357944 IC50 > 6000 nM T99685 C8IOD1 51357945 IC50 > 6000 nM T99685 C1KB9V 51357946 IC50 > 6000 nM T99685 C7HOD9 51357947 IC50 > 6000 nM T99685 CI7MJ6 51357948 IC50 > 6000 nM T99685 CRJ5W8 51358113 IC50 = 0.25 nM T99685 C9NS6B 52933960 IC50 = 41 nM T99685 CM24LF 52938983 IC50 = 3018 nM T99685 CU1P2L 52940797 IC50 = 100000 nM T99685 CD62QJ 52940982 IC50 = 93.5 nM T99685 C43SVQ 52941322 IC50 = 0.8 nM T99685 CK59HM 52941479 IC50 = 0.5 nM T99685 C3EJ9D 52941545 Ki = 947 nM T99685 C3ZOK1 52941683 Ki = 113 nM T99685 CDHJ08 52942235 IC50 = 10000 nM T99685 CHU8L6 52942777 Ki = 18 nM T99685 CFRN73 52942850 IC50 = 1.3 nM T99685 C4D1KT 52942879 IC50 = 3.45 nM T99685 C1XEV2 52943394 IC50 = 3600 nM T99685 C73WTL 52943744 IC50 = 1.1 nM T99685 C6Q1AH 52943745 IC50 = 1.85 nM T99685 CG7I1F 52943917 Ki = 6 nM T99685 CMG20V 52945133 Ki > 4000 nM T99685 CWD27C 52945142 IC50 = 0.73 nM T99685 CJ25NV 52945145 Ki = 3940 nM T99685 CWPC54 52945348 IC50 = 220 nM T99685 CXL53B 52945589 IC50 = 1.9 nM T99685 C4NLX7 52945630 IC50 = 2400 nM T99685 CXD6T8 52945845 IC50 = 16000 nM T99685 CN8F0V 52946289 IC50 = 13.5 nM T99685 CMQY93 52946368 IC50 = 1.55 nM T99685 C54LRW 52947235 IC50 = 1700 nM T99685 C5X9VO 52948007 IC50 = 3.3 nM T99685 CW9Z1T 52949347 IC50 = 2 nM T99685 CB0KM5 52949869 IC50 = 0.43 nM T99685 CE63PX 52949940 Ki = 5 nM T99685 CAJQ03 52950001 IC50 = 1.26 nM T99685 C5HQ2E 52950102 IC50 = 0.32 nM T99685 C4TNK8 52951283 IC50 = 1800 nM T99685 CJM04D 52951389 IC50 = 2500 nM T99685 C1VOS0 52951390 IC50 = 2100 nM T99685 CE05DT 53236130 Ki = 3 nM T99685 CP0L3O 53236131 Ki = 25 nM T99685 CD9WT7 53236132 Ki = 6 nM T99685 CG5BU3 53236606 Ki = 1.2 nM T99685 C6M0EG 53236607 Ki = 2.6 nM T99685 CFT4D9 53236823 Ki = 0.8 nM T99685 C5IFP3 53236824 Ki = 1.2 nM T99685 CDKV61 53237046 Ki = 1 nM T99685 CAL64M 53237047 Ki = 1.3 nM T99685 CJZ7I0 53237048 Ki = 0.34 nM T99685 C7QGN3 53237049 Ki = 0.66 nM T99685 CAS87Q 53237257 Ki = 4 nM T99685 C23VLY 53237258 Ki = 2.9 nM T99685 C6F5MH 53237259 Ki = 1 nM T99685 CR93EL 53237260 Ki = 1.1 nM T99685 COD8S4 53237261 Ki = 7 nM T99685 C6A3FN 53237262 Ki = 62 nM T99685 CYP5A7 53237477 Ki = 7.9 nM T99685 CIWE59 53237478 Ki = 1.7 nM T99685 CTM6D8 53237479 Ki = 6.8 nM T99685 C3Y8JZ 53237480 Ki = 21 nM T99685 CZ0LW2 53237719 Ki = 2.3 nM T99685 C34ZJA 53237720 Ki = 1.8 nM T99685 C39NBH 53237721 Ki = 3.2 nM T99685 CA85MY 53237722 Ki = 4.7 nM T99685 CT8IN1 53242225 IC50 = 600 nM T99685 C9NF0C 53302364 Ki = 8170 nM T99685 C4J9WZ 53307606 IC50 = 530 nM T99685 C7ZH0D 53308041 IC50 = 3.01 nM T99685 CT54XZ 53316658 Ki = 21 nM T99685 CG6O0M 53317018 Ki = 1330 nM T99685 C8FPQ4 53318293 Ki = 1000 nM T99685 CK9SE2 53318295 Ki = 84 nM T99685 CY8DH9 53322283 Ki = 1000 nM T99685 CN92LK 53322732 IC50 = 4000 nM T99685 CCSP27 53323641 Ki = 31 nM T99685 CW9F1T 53323642 Ki = 162 nM T99685 CQX59J 53323643 Ki = 216 nM T99685 CTD8A0 53324021 Ki = 3250 nM T99685 CZ41DR 53324923 Ki = 984 nM T99685 CZQ80X 53326214 Ki = 66 nM T99685 C25LHM 53326216 Ki = 17 nM T99685 CRYW35 53350231 Ki = 10 nM T99685 CCX7M5 53353847 Ki = 1260 nM T99685 C23HAU 53361718 IC50 = 1.6 nM T99685 CM60WQ 53361719 IC50 = 0.41 nM T99685 CBPR36 53363353 IC50 = 33 nM T99685 CL69DK 53377727 IC50 = 59 nM T99685 CG3C1J 53379513 IC50 = 0.7 nM T99685 C5SMC3 53387410 IC50 = 49 nM T99685 C5Q0HA 53387411 IC50 = 229 nM T99685 C90KZU 53387571 IC50 = 430 nM T99685 CMO9K1 53387572 IC50 = 446 nM T99685 CI40BG 53387573 IC50 = 70 nM T99685 C2IJR7 53387574 IC50 = 76 nM T99685 CWB79U 53387575 IC50 > 25000 nM T99685 CB4H9G 53387738 IC50 = 146 nM T99685 C5ZY9R 53387740 IC50 = 292 nM T99685 CVG90B 53389651 IC50 > 10000 nM T99685 CSV9X2 54579940 IC50 = 2 nM T99685 CN51TL 54579941 IC50 = 270 nM T99685 C7VZU2 54579942 IC50 = 260 nM T99685 C4R9JB 54579943 IC50 = 180 nM T99685 CG26HQ 54579944 IC50 = 80 nM T99685 CQE1Z7 54580062 IC50 = 390 nM T99685 C5O9WP 54580063 IC50 = 2100 nM T99685 CC5R3O 54580924 IC50 = 140 nM T99685 C3OIY4 54580925 IC50 = 45 nM T99685 CUP7N6 54581023 IC50 = 870 nM T99685 CAB63J 54581048 IC50 = 3000 nM T99685 C60TYL 54581049 IC50 = 190 nM T99685 CF2UH5 54581983 IC50 = 180 nM T99685 CB3OM9 54582056 IC50 = 3200 nM T99685 C5B4MV 54582091 IC50 = 110 nM T99685 C23EVN 54582916 IC50 = 680 nM T99685 CI8US3 54582917 IC50 = 33100 nM T99685 CT2SV7 54583916 IC50 = 175 nM T99685 CY87EC 54583917 IC50 = 680 nM T99685 C2GE8J 54584039 IC50 = 2400 nM T99685 C8CPI4 54584859 IC50 = 340 nM T99685 C9TZ2V 54584860 IC50 = 540 nM T99685 CVY42B 54584949 IC50 = 180 nM T99685 C1M9JE 54584986 IC50 = 1900 nM T99685 CME81Q 54585830 IC50 = 250 nM T99685 C81YUR 54585940 IC50 = 34 nM T99685 C1G0IY 54586917 IC50 = 4700 nM T99685 C0Y9ZG 54761473 IC50 = 150 nM T99685 CFUT05 56648675 Ki = 12 nM T99685 C1GAB6 56648677 Ki = 6.3 nM T99685 CWDF40 56648757 Ki = 14 nM T99685 CJO39U 56648759 Ki = 14 nM T99685 C83QGP 56660108 IC50 = 3 nM T99685 CYM1D0 56660109 IC50 = 0.3 nM T99685 CHA35L 56663573 IC50 = 18.5 nM T99685 CF7PY5 56667023 IC50 = 7.7 nM T99685 CC1DJ8 56670464 IC50 = 8.2 nM T99685 CZH95G 56673952 IC50 = 0.4 nM T99685 CHR8K0 56677282 IC50 = 5.6 nM T99685 C79AMB 56677283 IC50 = 22.5 nM T99685 C5ZN6X 56682067 IC50 = 24 nM T99685 CG17TZ 56683916 IC50 = 14.5 nM T99685 C7B2OH 56683917 IC50 = 1.1 nM T99685 C6LMP8 56683918 IC50 = 1.7 nM T99685 C94JIT 56832510 IC50 > 4300 nM T99685 C4Z0OC 56834890 Ki = 2800 nM T99685 C67TJQ 56834891 Ki = 2600 nM T99685 C32CID 56926598 Ki = 3900 nM T99685 CV8Z5C 56926697 Ki = 3900 nM T99685 CO43FQ 56926699 Ki = 1100 nM T99685 C4GT2U 56926701 Ki = 2100 nM T99685 CPGC81 56947516 IC50 > 10000 nM T99685 C0M3EQ 56950791 IC50 = 84 nM T99685 CAK91L 56955954 IC50 = 623 nM T99685 C74YNV 56966983 IC50 = 751 nM T99685 CVK5A3 57328247 IC50 > 10000 nM T99685 CZ7RE0 57345686 IC50 = 32000 nM T99685 C3CL8H 57384862 Ki = 1200 nM T99685 C96WSJ 57387650 Ki = 13 nM T99685 C6I8SF 57390697 IC50 = 3500 nM T99685 C3R2LD 57390793 IC50 = 1590 nM T99685 C9RB7K 57391333 IC50 > 10000 nM T99685 CH37SE 57391335 IC50 > 10000 nM T99685 C0QF7X 57392605 IC50 = 9 nM T99685 C8U6ZC 57392648 IC50 = 120 nM T99685 C7XS2P 57394206 IC50 = 30 nM T99685 CFG53Z 57394325 IC50 > 10000 nM T99685 CSRG42 57394326 IC50 = 2020 nM T99685 C45NDO 57394361 IC50 = 8300 nM T99685 C09MPI 57396034 IC50 = 170 nM T99685 CA52UR 57396083 IC50 = 8900 nM T99685 CS14ZH 57396608 IC50 > 10000 nM T99685 CLJ5B1 57397772 IC50 = 2 nM T99685 C4N7MX 57397773 IC50 = 6 nM T99685 C2XZG9 57397841 IC50 = 390 nM T99685 C2VPR0 57397894 IC50 = 30 nM T99685 CU9N1Z 57398248 IC50 = 71 nM T99685 CQO74C 57398382 IC50 > 10000 nM T99685 CV2Z0C 57398383 IC50 > 10000 nM T99685 C9Z6AL 57399433 IC50 = 10 nM T99685 CA3NV0 57399544 IC50 = 9 nM T99685 C7UYA9 57401258 IC50 = 120 nM T99685 CJC26L 57401330 IC50 > 10000 nM T99685 C0LP7R 57401331 IC50 = 70 nM T99685 CRO5Z6 57401846 IC50 > 10000 nM T99685 CWV56Z 57402952 IC50 = 63 nM T99685 C5TPX8 57403086 IC50 = 130 nM T99685 C8Y7VZ 57427751 IC50 = 758.58 nM T99685 CK6TN2 57427752 IC50 = 5.754 nM T99685 CT6XL0 57466811 IC50 > 9100 nM T99685 C59YAC 57495353 IC50 > 9100 nM T99685 CWQ6F2 57523291 IC50 > 10000 nM T99685 CJE19S 57523686 IC50 > 10000 nM T99685 C1EP6I 58024825 IC50 = 2600 nM T99685 CX8SZ7 58118657 IC50 < 31.62 nM T99685 C46AUK 58137055 IC50 = 262 nM T99685 C7ONC3 58137106 IC50 = 330 nM T99685 C6DH9J 58137111 IC50 = 3160 nM T99685 C7VSX2 58137137 IC50 = 601 nM T99685 C84FUI 58137148 IC50 = 1540 nM T99685 C5IMD7 58137170 IC50 = 1380 nM T99685 CRPL37 58137176 IC50 = 285 nM T99685 CV7YP2 58169819 IC50 = 7.943 nM T99685 CJ8TE4 58169820 IC50 = 12.59 nM T99685 CU3WG8 58298312 IC50 = 106 nM T99685 CONJ64 58298326 IC50 = 30 nM T99685 C0W7QE 58298327 IC50 = 19 nM T99685 C7GIQ1 58298333 IC50 = 175 nM T99685 CB9XN5 58298334 IC50 = 66 nM T99685 C7GA2Y 58379501 Ki = 0.243 nM T99685 C0D7NE 58379507 Ki = 0.842 nM T99685 CO5NX4 58379530 Ki = 18.5 nM T99685 CVL1G3 58379533 Ki = 2.64 nM T99685 C2DM7X 58379543 Ki = 2.2 nM T99685 C5YQL3 58379551 Ki = 2.33 nM T99685 CX01MF 58379559 Ki = 4.71 nM T99685 CT9W7U 58379595 Ki = 1.55 nM T99685 CFE09U 58379619 Ki = 2 nM T99685 C31NXY 58379638 Ki = 47.4 nM T99685 CUTJ73 58379663 Ki = 0.377 nM T99685 CZUO79 58441681 IC50 = 0.75 nM T99685 CB2VP8 58507929 Ki = 19.3 nM T99685 CK0O4B 58508043 Ki = 109 nM T99685 C1I4ZO 58508110 Ki = 64.5 nM T99685 CPCG46 58508197 Ki = 224 nM T99685 C85HOT 58508283 Ki = 25.5 nM T99685 C58FIX 58508310 Ki = 609 nM T99685 CBA73C 59239059 Ki = 48 nM T99685 CDM57O 59239077 Ki = 2.4 nM T99685 C0XN3Y 59239089 Ki = 6.5 nM T99685 CQ4HD1 59239114 Ki = 1.5 nM T99685 CY3M0Z 59239164 Ki = 1.7 nM T99685 C18DJR 59239174 Ki = 6.8 nM T99685 CYOW74 59239188 Ki = 20 nM T99685 C42ZDM 59239194 Ki = 2.4 nM T99685 CRKP62 59239206 Ki = 3 nM T99685 CM0AY7 59239207 Ki = 4.2 nM T99685 CG1A8Y 59239249 Ki = 1.3 nM T99685 COEM65 59239271 Ki = 220 nM T99685 CIR81P 59239300 Ki = 0.4 nM T99685 C82YHL 59239336 Ki = 11 nM T99685 C6MQA3 59239348 Ki = 1.4 nM T99685 CN9WD1 59239356 Ki = 2.3 nM T99685 C6ZRI4 59239369 Ki = 5.5 nM T99685 C2BX0H 59239374 Ki = 18 nM T99685 CQ6I7T 59239380 Ki = 130 nM T99685 CP64KI 59239424 Ki = 2.7 nM T99685 CVG8B3 59239456 Ki = 3.5 nM T99685 CTX01P 59239521 Ki = 2.7 nM T99685 C4YW3N 59239622 Ki = 3.7 nM T99685 CDX4G0 59258834 Ki = 51.2 nM T99685 CY0SB7 59258852 Ki = 76.4 nM T99685 CSJ60G 59258855 Ki = 23.5 nM T99685 CSIV71 59258894 Ki = 110 nM T99685 CCZ9F4 59258904 Ki = 700 nM T99685 C36ZSD 59258941 Ki = 10.6 nM T99685 CJ4ME2 59258944 Ki = 190 nM T99685 C4SRU6 59258964 Ki = 18.6 nM T99685 COA89E 59258965 Ki = 82 nM T99685 CUF6Y9 59259010 Ki = 150 nM T99685 CD43UI 59259014 Ki = 272 nM T99685 C3NKS2 59259019 IC50 = 30.09 nM T99685 CI2SU0 59453028 IC50 = 8 nM T99685 CY8L4O 59453029 IC50 = 12 nM T99685 CTMA05 59453047 IC50 = 14 nM T99685 C8YDC3 59453057 IC50 = 103 nM T99685 CYN1L2 59453060 IC50 = 103 nM T99685 CA4XV9 59453066 IC50 = 25 nM T99685 C1I7QA 59453069 IC50 = 5 nM T99685 CNV0I9 59453076 IC50 = 38 nM T99685 CQYI53 59453077 IC50 = 12 nM T99685 CV6A4J 59453078 IC50 = 8 nM T99685 CM2Q5J 59453081 IC50 = 3 nM T99685 CV1SY9 59453083 IC50 = 185 nM T99685 CPH5N4 59453087 IC50 = 436 nM T99685 CRFC53 59453089 IC50 = 15 nM T99685 C1RTQ6 59453093 IC50 = 33 nM T99685 C26QRA 59453105 IC50 = 37 nM T99685 C2BM8E 59453110 IC50 = 26 nM T99685 C0WQ4N 59453111 IC50 = 4 nM T99685 CO9G5I 59453117 IC50 = 72 nM T99685 CWJ3L7 59453121 IC50 = 4 nM T99685 CLQ08G 59453125 IC50 = 168 nM T99685 CXA9D8 59453133 IC50 = 46 nM T99685 C5D6ZW 59477194 IC50 = 385 nM T99685 C2X8TY 59548177 IC50 > 10000 nM T99685 C71GBC 59548184 IC50 > 10000 nM T99685 C10NEZ 59548195 IC50 > 25000 nM T99685 CGRO45 59548196 IC50 > 10000 nM T99685 CD39AG 59548207 IC50 > 10000 nM T99685 C5B0MY 59548213 IC50 = 10600 nM T99685 C6KP4G 59548220 IC50 > 10000 nM T99685 CL82RM 59548221 IC50 > 10000 nM T99685 CTNU85 59548226 IC50 > 10000 nM T99685 CLF4I3 59548231 IC50 = 6700 nM T99685 CLB6N4 59548232 IC50 = 5100 nM T99685 C2KBG8 59548236 IC50 > 10000 nM T99685 CSWV07 59548243 IC50 > 10000 nM T99685 CN48VL 59548245 IC50 > 10000 nM T99685 CMT2R0 59548250 IC50 > 10000 nM T99685 CT5RK1 59548255 IC50 > 16000 nM T99685 C3I8NE 59548256 IC50 > 10000 nM T99685 C8W5HT 59548263 IC50 > 10000 nM T99685 C4WOJ7 59548265 IC50 = 2500 nM T99685 CT8Q5B 59548274 IC50 > 10000 nM T99685 C8FSH7 59548276 IC50 = 2100 nM T99685 CBG52T 59548278 IC50 > 10000 nM T99685 CVF1B2 59548283 IC50 > 10000 nM T99685 CY31EA 59548284 IC50 > 10000 nM T99685 CO4GT7 59548288 IC50 = 163 nM T99685 CFR7S8 59548302 IC50 = 2500 nM T99685 CRE8B3 59548316 IC50 > 10000 nM T99685 C7I9QW 59548318 IC50 = 3700 nM T99685 CRM20Z 59548320 IC50 > 10000 nM T99685 CX1KJ9 59548322 IC50 > 10000 nM T99685 CJE5I4 59548341 IC50 > 10000 nM T99685 CSFV40 59548348 IC50 = 2200 nM T99685 C8O1VS 59548349 IC50 = 3600 nM T99685 CE9W0K 59548355 IC50 > 10000 nM T99685 CWC65A 59548356 IC50 > 10000 nM T99685 CMKP95 59548371 IC50 > 10000 nM T99685 C72TQL 59548376 IC50 > 22000 nM T99685 CC8UV3 59548383 IC50 = 290 nM T99685 CK7ZS8 59548389 IC50 > 17000 nM T99685 C4SN3U 59548390 IC50 > 10000 nM T99685 C5O3BM 59548393 IC50 = 7800 nM T99685 CD4ET2 59548402 IC50 > 10000 nM T99685 CES59T 59548403 IC50 > 10000 nM T99685 CE8P3G 59548407 IC50 = 32 nM T99685 CO4K2W 59548419 IC50 = 74 nM T99685 CSDB78 59548424 IC50 > 10000 nM T99685 C81FCQ 59548431 IC50 > 10000 nM T99685 CLGY34 59548453 IC50 > 10000 nM T99685 CBT21W 59548454 IC50 > 10000 nM T99685 C9DIB3 59548458 IC50 > 10000 nM T99685 CJT68K 59548460 IC50 > 10000 nM T99685 C9LFT3 59548462 IC50 > 10000 nM T99685 C6PVN9 59548463 IC50 = 7800 nM T99685 CA47YQ 59548474 IC50 > 10000 nM T99685 CX8C2U 59548480 IC50 > 10000 nM T99685 CM8PD7 60150509 IC50 = 6300 nM T99685 C5KD3Z 60154714 IC50 > 10000 nM T99685 CS0L4D 60154996 IC50 > 10000 nM T99685 C1UI3P 60155086 IC50 > 10000 nM T99685 CX08ON 60155087 IC50 > 10000 nM T99685 CX8J1I 60155265 IC50 > 10000 nM T99685 CAT40I 60155266 IC50 > 10000 nM T99685 CD56VA 60155268 IC50 = 1400 nM T99685 C5FI4P 60155451 IC50 = 3700 nM T99685 CX9G4U 60155452 IC50 = 1400 nM T99685 CR7EG9 60155538 IC50 > 10000 nM T99685 CU6YB9 60155539 IC50 > 10000 nM T99685 CSZA16 60155724 IC50 = 1781 nM T99685 C6BY2S 60210977 IC50 = 890 nM T99685 C6GE5S 62705166 Ki = 663 nM T99685 C94MTA 62705167 Ki = 123 nM T99685 CV0MD4 62705168 Ki = 13 nM T99685 CSD3F8 62705169 Ki = 15 nM T99685 C3LS8Q 62705170 Ki = 52 nM T99685 C2E3AO 62705171 IC50 = 6 nM T99685 CSD0N6 62705990 IC50 = 15 nM T99685 C9NI6K 62705991 IC50 = 27 nM T99685 C2RDA4 62706154 IC50 = 6 nM T99685 C3M6QC 62706155 IC50 = 3 nM T99685 CAG23H 62706156 IC50 = 3 nM T99685 C1RB8F 62706157 IC50 = 21 nM T99685 CGC62F 62706158 IC50 = 2 nM T99685 C67TAB 62706159 IC50 = 39 nM T99685 C4IGR0 62706312 IC50 = 4 nM T99685 CPM5R9 62706313 IC50 = 2 nM T99685 CX6IU3 62706314 IC50 = 3 nM T99685 CFJ8W5 62706315 IC50 = 10 nM T99685 CX0H7E 62706316 IC50 = 5 nM T99685 C06IUA 62706317 IC50 = 2 nM T99685 C82NPI 62706470 IC50 = 3 nM T99685 CPR50J 62706471 IC50 = 76 nM T99685 CA31ZB 62706472 IC50 = 65 nM T99685 CWRJ86 62706475 IC50 = 63 nM T99685 CNMX21 62706476 IC50 = 141 nM T99685 CS0CA6 62706650 IC50 = 3 nM T99685 C71APZ 62706651 IC50 = 6 nM T99685 CFBD83 62706652 IC50 = 147 nM T99685 CL20FV 62706653 IC50 = 24 nM T99685 C34MPU 62706654 IC50 = 36 nM T99685 CHX01T 62706655 IC50 = 55 nM T99685 CM39TP 62706813 IC50 = 9 nM T99685 CHK4I1 62706814 IC50 = 67 nM T99685 C16ZGX 62706815 IC50 = 15 nM T99685 CS4VA8 62706816 IC50 = 16 nM T99685 CY0D8M 62706817 IC50 = 20 nM T99685 C9G5NA 62707451 Ki = 25 nM T99685 CWZ1I7 62707452 Ki = 50 nM T99685 C7ZY3Q 62707454 Ki = 120 nM T99685 C80KUA 62707599 Ki = 5 nM T99685 C9RV1U 62707603 Ki = 7 nM T99685 CU2P1Z 62707604 Ki = 62 nM T99685 CUC7B3 66557964 IC50 = 42000 nM T99685 CWZ54O 66600540 IC50 > 10000 nM T99685 C6Q0KU 66612050 IC50 > 10000 nM T99685 C0X9FR 66699750 IC50 = 2 nM T99685 CB8WP9 66788776 IC50 = 34 nM T99685 C51ARE 66788835 IC50 = 206 nM T99685 C6DYG9 66788911 IC50 = 412 nM T99685 CQ5TC4 66789238 IC50 = 20 nM T99685 CIR86Z 66789609 IC50 = 57 nM T99685 CYKD92 66789704 IC50 = 36 nM T99685 CRO34N 66790135 IC50 = 157 nM T99685 COE7X1 66790311 IC50 = 12 nM T99685 CUJB72 66790335 IC50 = 62 nM T99685 CU58AM 67073110 Ki = 2470 nM T99685 C1K5PQ 67094257 Ki = 8 nM T99685 CJ46YU 67094333 Ki = 12 nM T99685 CT9AH0 67178880 Ki = 3.2 nM T99685 CIT38E 67179786 Ki = 4.4 nM T99685 CA1WS0 67276196 Ki = 1.4 nM T99685 C4MX9K 67276455 Ki = 4.8 nM T99685 C9LI0M 67294297 Ki = 1700 nM T99685 C1HBC0 67535197 IC50 = 1.7 nM T99685 CNZ2C3 67535447 IC50 = 277 nM T99685 C3M1OJ 67535551 IC50 = 16 nM T99685 C97SXL 68194826 IC50 = 316.23 nM T99685 CJ2BU0 68195106 IC50 > 2000 nM T99685 C3VKM5 68512988 IC50 > 15000 nM T99685 C2D4BQ 68518711 IC50 = 11100 nM T99685 CC63RO 68893189 IC50 = 2 nM T99685 C45TIJ 69489467 IC50 = 1260 nM T99685 CNX20F 70676303 Ki = 9 nM T99685 CM8H3V 70676450 Ki = 21 nM T99685 CDMO03 70682114 IC50 = 2290 nM T99685 C65LPD 70684413 Ki = 50 nM T99685 CG95EC 70684794 IC50 = 5710 nM T99685 CQS8G7 70686830 IC50 > 9100 nM T99685 CMC74I 70688479 IC50 > 5000 nM T99685 CQ04ZJ 70689027 IC50 = 5100 nM T99685 CN45VU 70690535 IC50 > 5000 nM T99685 CC64RD 70692128 IC50 = 22500 nM T99685 C7ASK8 70692129 IC50 = 252 nM T99685 CU3WF2 70693248 IC50 = 10000000 nM T99685 C4P9CL 70693798 Ki = 434 nM T99685 CX2JZ1 70694178 IC50 > 100000 nM T99685 C7HW2B 70694179 IC50 = 37 nM T99685 CICE82 70694721 IC50 > 5000 nM T99685 C38LWS 70694722 IC50 > 5000 nM T99685 CLY5G3 70695401 IC50 > 30000 nM T99685 CF8EK2 71250848 IC50 = 32 nM T99685 CJP69K 71250855 IC50 = 146 nM T99685 C8KD6L 71250859 IC50 = 95 nM T99685 CM10HY 71250872 IC50 = 72 nM T99685 CS3V1R 71250875 IC50 > 500 nM T99685 C85IZO 71250882 IC50 = 48 nM T99685 C1LI6X 71250891 IC50 = 2 nM T99685 CSO29K 71250896 IC50 = 30 nM T99685 CKE7H2 71250907 IC50 = 88 nM T99685 CI5MT1 71250909 IC50 > 500 nM T99685 C9G2MT 71250929 IC50 = 10 nM T99685 CZP1E8 71250935 IC50 = 53 nM T99685 C1MVL0 71273460 Ki = 1840 nM T99685 C6SAW5 71449586 IC50 > 20000 nM T99685 CK58RV 71449587 IC50 = 18 nM T99685 C6GJE3 71451395 IC50 = 4600 nM T99685 CD8Y3S 71451617 IC50 > 10000 nM T99685 C5KH7C 71453205 IC50 = 16 nM T99685 C6VF7J 71453206 IC50 = 18 nM T99685 CR84JX 71453419 IC50 = 7 nM T99685 CZ8Q5P 71454238 IC50 = 198 nM T99685 CO0WF5 71454941 IC50 = 610 nM T99685 CA30GO 71454942 IC50 = 1700 nM T99685 CH3WN6 71454943 IC50 > 4000 nM T99685 CF74SL 71454944 IC50 = 88 nM T99685 CO82IY 71455167 IC50 > 10000 nM T99685 CA7L1Y 71455168 IC50 > 10000 nM T99685 COW5S1 71456726 IC50 = 3300 nM T99685 CZG8I6 71456727 IC50 = 140 nM T99685 CE1IX7 71456728 IC50 = 25 nM T99685 C14OGU 71458568 IC50 = 320 nM T99685 C6CR7L 71458569 IC50 > 20000 nM T99685 CWAU20 71458570 IC50 > 4000 nM T99685 CVQ62G 71458571 IC50 = 110 nM T99685 C74VKX 71458572 IC50 = 3200 nM T99685 CM1ND2 71458573 IC50 = 15 nM T99685 C3S0NP 71458574 IC50 = 45 nM T99685 CY6WI2 71458575 IC50 = 50 nM T99685 C15XAV 71460420 IC50 = 200 nM T99685 CKV1P2 71460421 IC50 = 7.7 nM T99685 CT7K3A 71460422 IC50 = 12 nM T99685 C25FQP 71462104 IC50 > 20000 nM T99685 CY74CX 71472903 IC50 = 16620 nM T99685 CB78IN 71493938 IC50 = 29 nM T99685 CV03AL 71541406 Ki = 13.4 nM T99685 C7V9SQ 71547699 IC50 = 226 nM T99685 CBCW18 71571355 Ki = 8.63 nM T99685 CQ16UM 71584055 IC50 = 190 nM T99685 C1GDL2 71602514 Ki = 12.8 nM T99685 CHV4N8 71602515 Ki = 24.4 nM T99685 C7YVU4 71602573 Ki = 4.46 nM T99685 C90PSW 71602574 Ki = 2.15 nM T99685 C34HNA 71602575 Ki = 19.5 nM T99685 CM06KQ 71602576 Ki = 7.82 nM T99685 COG0X5 71604742 Ki = 4.2 nM T99685 CC5UR3 71604893 Ki = 4.2 nM T99685 COZ4A6 71604894 Ki = 6.5 nM T99685 C13FGZ 71604895 Ki = 14 nM T99685 C4NA0Z 71604896 Ki = 21 nM T99685 CNY35F 71604897 Ki = 2.6 nM T99685 CN08ZO 71605054 Ki = 7.5 nM T99685 CHK8Y6 71605056 Ki = 6.5 nM T99685 C0HEN3 71605057 Ki = 1.2 nM T99685 C2FAE3 71716356 IC50 = 1300 nM T99685 C5K9JV 71717638 Ki = 0.99 nM T99685 C5S8DT 71717639 Ki = 1.2 nM T99685 CJP83B 71719453 Ki = 1.2 nM T99685 C86MQI 71720046 Ki = 1.5 nM T99685 CLT60U 71720047 Ki = 2.1 nM T99685 C7EY1Q 72163951 Ki = 9 nM T99685 CVT76M 72163952 Ki = 7 nM T99685 C9UOH5 72164062 Ki = 6 nM T99685 CT3X8G 72164184 Ki = 19 nM T99685 CLO1P5 72199292 IC50 = 0.6 nM T99685 C9E4XZ 72546233 IC50 > 3000 nM T99685 C29KOU 72709209 IC50 > 10000 nM T99685 CT73IW 72709284 IC50 > 10000 nM T99685 CW6V2I 72947132 IC50 > 2000 nM T99685 CWL0F2 73054768 IC50 = 67 nM T99685 C95YFI 73054769 IC50 = 62 nM T99685 C8EI1X 73673707 IC50 = 3.8 nM T99685 CBYN18 73977439 IC50 = 1622 nM T99685 C9V1YR 73977449 IC50 = 468 nM T99685 CXA90D 73977451 IC50 = 380 nM T99685 CEZ7L2 73977461 IC50 = 1175 nM T99685 CD0T9V 74539799 IC50 = 1.1 nM T99685 C16KOS 74539862 IC50 = 2.2 nM T99685 CKO41J 76310248 IC50 = 100 nM T99685 CEN9Q5 76310249 IC50 = 127 nM T99685 CJCF67 76310250 IC50 = 5 nM T99685 CBI09O 76310352 IC50 = 8.49 nM T99685 CMF0R5 76310353 IC50 = 28.68 nM T99685 C06OME 76310354 IC50 = 62.64 nM T99685 C4BT9H 76314027 IC50 = 125.93 nM T99685 CC8NB4 76314028 IC50 = 18.39 nM T99685 C4MKN3 76317469 IC50 = 1 nM T99685 C3JA4F 76317470 IC50 = 36 nM T99685 C3XYV1 76317571 IC50 = 12.25 nM T99685 CPK6B4 76317572 IC50 = 65.64 nM T99685 C8E4GI 76321204 IC50 = 336 nM T99685 CPLO52 76321296 IC50 = 13.36 nM T99685 CGY1N5 76321297 IC50 > 10000 nM T99685 C34OYK 76321298 IC50 = 35.27 nM T99685 CE35LN 76321299 IC50 = 36.54 nM T99685 CDG8V4 76324821 IC50 = 266 nM T99685 C2BFA1 76324823 IC50 = 400 nM T99685 CZTR31 76324910 IC50 = 35.02 nM T99685 C4FMR8 76324911 IC50 = 13.88 nM T99685 C8X9TV 76324913 IC50 = 11.19 nM T99685 CX3N7R 76328473 IC50 = 2.32 nM T99685 CE5I7T 76328474 IC50 = 39.04 nM T99685 CUC04I 76328475 IC50 = 140.9 nM T99685 C70WJE 76332052 IC50 = 35 nM T99685 CKD7H2 76332159 IC50 > 10000 nM T99685 C8SL3V 76332160 IC50 = 82.12 nM T99685 C3KIG0 76332161 IC50 = 33.92 nM T99685 CZ92PW 76335665 IC50 = 453 nM T99685 C73KJD 76335670 IC50 = 13 nM T99685 CD2KU1 76335780 IC50 = 78.2 nM T99685 C47ZNT 76335781 IC50 = 159.96 nM T99685 CSCK18 76335782 IC50 = 13.91 nM T99685 CRD94L 76335783 IC50 = 171.72 nM T99685 C6VCF1 76335784 IC50 = 8.55 nM T99685 CT1UL6 76335785 IC50 = 19.2 nM T99685 CU86DF 76335786 IC50 = 24.69 nM T99685 C2JTH8 77107528 IC50 > 1000 nM T99685 C42HDP 77107927 IC50 = 580 nM T99685 C04SRC 77147259 IC50 = 1060 nM T99685 C37LKW 86346018 IC50 = 1100 nM T99685 CK8XE9 86652633 IC50 = 328 nM T99685 CNVS32 87343636 Ki = 5410 nM T99685 CB1VI6 90665817 Ki = 16 nM T99685 CP1W6K 91755004 IC50 = 45.8 nM T99685 C64QBH 117995822 Ki = 69 nM T99685 C7KTW4 118000035 Ki = 812 nM T99685 C7E2DY 118000150 Ki = 24 nM T99685 CKZ5N0 118000206 Ki = 1279 nM T99685 C72IRG 118321317 IC50 = 37.6 nM T99685 C7EAJ0 118321318 IC50 = 245 nM T99685 C8AR0W 118321320 IC50 = 79.2 nM T99685 CBE08T 118321322 IC50 = 180 nM T99685 C67XRL 118321324 IC50 = 111 nM T99685 CH7MG0 118321327 IC50 = 67 nM T99685 C1H7SU 118470918 Ki = 284 nM T99685 CM2DO8 118616331 IC50 = 138 nM T99685 CO0YC8 118616775 IC50 = 89.2 nM T99685 C42SYZ 118616923 IC50 = 197.9 nM T99685 CXA8N2 118616927 IC50 = 105.8 nM T99685 C84DGB 118616929 IC50 > 400 nM T99685 C8SRG9 118616951 IC50 = 64 nM T99685 CFQ71C 118616958 IC50 = 108.5 nM T99685 CU6E0P 118616985 IC50 > 400 nM T99685 C7WO2R 118617086 IC50 > 400 nM T99685 CVJU09 118617088 IC50 = 245.7 nM T99685 CQ7A1G 118617093 IC50 = 163.3 nM T99685 C6U0GQ 118617094 IC50 = 153.4 nM T99685 CB5XL3 118617097 IC50 = 223.4 nM T99685 CZ30BK 118617099 IC50 = 119 nM T99685 CGVH36 118617158 IC50 = 66 nM T99685 C4AHL2 118711367 IC50 > 10000 nM T99685 CF5HV8 118720613 IC50 = 1100 nM T99685 C2UIB7 118720614 IC50 > 2300 nM T99685 CSH50J 118720615 IC50 = 4400 nM T99685 C4LW6I 118720885 IC50 > 4600 nM T99685 C9Y4EH 118720886 IC50 = 7500 nM T99685 C9SF2E 118720891 IC50 > 13000 nM T99685 CQV64Y 118722479 IC50 > 15000 nM T99685 CDLC32 118722480 IC50 > 25000 nM T99685 CP9QZ8 118722481 IC50 > 25000 nM T99685 C8Y2AF 118722482 IC50 = 790 nM T99685 C39TEL 118722483 IC50 = 15800 nM T99685 CM4Q5D 118722770 IC50 > 25000 nM T99685 CQCX41 118737057 IC50 > 10000 nM T99685 CKBP72 121231408 IC50 > 10000 nM T99685 CK0LZ1 121275690 IC50 = 1.6 nM T99685 CIN39H 121334370 Ki = 192 nM T99685 CJDS80 121334379 Ki = 12.6 nM T99685 CC1R8L 121334382 Ki = 650 nM T99685 CU37QN 121334400 Ki = 31 nM T99685 CSKB71 121334407 Ki = 73.4 nM T99685 CM2ZS6 121334410 Ki = 60.2 nM T99685 C4R7DN 121334420 Ki = 42.3 nM T99685 CK3G6P 121334425 Ki = 10 nM T99685 C01CNO 121334433 Ki = 7.4 nM T99685 CGCL96 121334436 Ki = 15.3 nM T99685 CB1L6S 121334438 Ki = 42 nM T99685 CV92TK 121334444 Ki = 35 nM T99685 CGD9K5 121334446 Ki = 11.2 nM T99685 CYTA71 121334474 Ki = 3.5 nM T99685 CH6Y9L 121334475 Ki = 13.9 nM T99685 CHX60O 121334481 Ki = 12 nM T99685 CYI09J 121334494 Ki = 13.6 nM T99685 CZ46TQ 121334504 Ki = 10.6 nM T99685 COZT28 121334509 Ki = 6.9 nM T99685 C1YQ8R 121334511 Ki = 32.8 nM T99685 C8M2ET 121334520 Ki = 10.8 nM T99685 C91PVZ 121428416 IC50 = 186 nM T99685 CA2DM0 121428489 IC50 = 2120 nM T99685 CQLX36 121428567 IC50 = 1680 nM T99685 CI1PS7 121428640 IC50 = 13980 nM T99685 C81IFQ 122163152 IC50 = 15 nM T99685 CL36RB 122178108 IC50 = 66.7 nM T99685 C4Q5KS 122178109 IC50 = 3.04 nM T99685 C2BV9G 122178110 IC50 = 0.2 nM T99685 CCHI06 122178111 IC50 = 62.3 nM T99685 C3FS4U 122178112 IC50 = 21.6 nM T99685 CT5J4A 122178113 IC50 = 0.29 nM T99685 C2VGD5 122178120 IC50 = 218 nM T99685 CTE0F7 122178121 IC50 = 363 nM T99685 C3S2UI 122178122 IC50 = 67.9 nM T99685 C57MXE 122178123 IC50 = 345 nM T99685 C24XUZ 122178124 IC50 = 53.6 nM T99685 C3XMW0 122178125 IC50 = 43.7 nM T99685 C2P6KC 122178126 IC50 = 25.8 nM T99685 CS85CU 122181413 IC50 = 15000 nM T99685 CQS67B 122181416 IC50 = 21000 nM T99685 C0NJ3A 122182356 IC50 = 613 nM T99685 CKT74G 122185265 IC50 = 275 nM T99685 CJ6C1O 122185267 IC50 = 123 nM T99685 CD67LU 122705248 IC50 = 8565 nM T99685 CX63VW 122705258 IC50 > 10000 nM T99685 C76IKM 122705261 IC50 = 328 nM T99685 C8ALO2 124088839 IC50 > 10000 nM T99685 C98DKI 127025346 IC50 = 9.9 nM T99685 CBXJ67 127025628 IC50 = 5.4 nM T99685 CB53ZX 127028515 IC50 = 860 nM T99685 CB9VY8 127028516 IC50 = 940 nM T99685 CSV3R7 127029064 IC50 = 78 nM T99685 CAD38Y 127029440 IC50 = 9430 nM T99685 CR17GV 127029715 IC50 = 6260 nM T99685 CQV05N 127032901 IC50 = 114 nM T99685 C0S5WG 127032910 IC50 = 46 nM T99685 CH7QO2 127032911 IC50 = 17 nM T99685 CNA82D 127032912 IC50 > 3000 nM T99685 CMD0Z8 127032913 IC50 > 3000 nM T99685 C59RLZ 127032914 IC50 > 3000 nM T99685 CGKR53 127032915 IC50 = 30 nM T99685 CT3R6Y 127033229 IC50 = 22 nM T99685 CYNX65 127033230 IC50 = 340 nM T99685 CY8UZ1 127033231 IC50 = 310 nM T99685 CKT2Q6 127034306 IC50 = 25 nM T99685 CEF18H 127034307 IC50 = 36 nM T99685 CY1TR5 127035128 IC50 = 1105 nM T99685 CQTE98 127035129 IC50 = 33 nM T99685 CV94GA 127035130 IC50 = 514 nM T99685 CWUK71 127035185 IC50 = 73 nM T99685 C2ZJA9 127035281 IC50 = 30 nM T99685 CW0I4F 127035282 IC50 = 280 nM T99685 CQ3BK8 127035283 IC50 = 674 nM T99685 CJ2E4N 127035335 IC50 = 21 nM T99685 CM9UL5 127035423 IC50 = 51 nM T99685 C7G8JM 127035424 IC50 = 361 nM T99685 CBV03O 127035425 IC50 = 14 nM T99685 CI6D9M 127035790 IC50 = 806 nM T99685 C5ICR3 127035792 IC50 > 3000 nM T99685 C8PO0M 127035794 IC50 = 284 nM T99685 CJK1X6 127035909 IC50 = 24 nM T99685 CZWA79 127035980 IC50 = 1225 nM T99685 C41YQI 127035981 IC50 = 31 nM T99685 CG8DA9 127045861 IC50 = 25 nM T99685 CVF8Z9 127045862 IC50 = 1.8 nM T99685 CH68NT 127046076 IC50 = 5 nM T99685 CA2XD5 127046077 IC50 = 1 nM T99685 C34REM 127046317 IC50 > 50000 nM T99685 CC4ND8 127046862 IC50 = 59 nM T99685 CO25WH 127052538 IC50 > 10000 nM T99685 CK68CA 130453737 IC50 = 21000 nM T99685 CUO41K 130470684 IC50 = 1480 nM T99685 CBY49C 132156028 Ki = 9.6 nM T99685 CPZ02V 132563118 IC50 = 114 nM T99685 C21KNJ 132563119 IC50 = 208 nM T99685 CT2PN8 132990561 IC50 = 16 nM T99685 C2AN7T 134611886 IC50 > 100000 nM T99685 CX0UR7 134694318 IC50 = 2920 nM T99685 C54FXD 134957362 IC50 > 10000 nM T99685 CT0GQ6 135197577 IC50 = 43 nM T99685 C87VKA 135197594 IC50 = 56 nM T99685 CQXS07 135197635 IC50 = 9.9 nM T99685 C7KXF1 135197643 IC50 = 7.9 nM T99685 CEK31P 135566415 IC50 > 20000 nM T99685 C24ZGX 135566644 IC50 > 10000 nM T99685 C2QDV5 135566741 IC50 > 10000 nM T99685 CU29YK 135750268 IC50 = 6000 nM T99685 CD6UJ5 135857414 IC50 = 1265 nM T99685 C41HNJ 135857415 IC50 = 170 nM T99685 CX4ZB3 135863110 IC50 = 18000 nM T99685 CRFO90 135870998 IC50 = 1020 nM T99685 CZ7Y0P 135871000 IC50 = 2880 nM T99685 C8K3HJ 135911704 IC50 = 23 nM T99685 C12UDA 135947972 IC50 = 3 nM T99685 CN42ZS 135947973 IC50 = 2100 nM T99685 CF8AO3 135947974 IC50 = 1130 nM T99685 CW08GJ 135947976 IC50 = 20 nM T99685 CJN7E2 135947978 IC50 = 1200 nM T99685 CFKH34 135947979 IC50 = 109 nM T99685 CXH63V 136041747 IC50 > 10000 nM T99685 C6B5TC 136041748 IC50 > 10000 nM T99685 CU6XG1 136041749 IC50 > 10000 nM T99685 C0U5DB 136041750 IC50 > 10000 nM T99685 C48KAQ 136041752 IC50 > 10000 nM T99685 C74PRL 136041753 IC50 > 10000 nM T99685 CCS2G6 136041761 IC50 > 10000 nM T99685 CEZP21 136041762 IC50 > 10000 nM T99685 CJ58TD 136041764 IC50 > 10000 nM T99685 CX67QW 136041765 IC50 > 10000 nM T99685 CK0H2Q 136041766 IC50 > 10000 nM T99685 CM65BS 136041773 IC50 > 10000 nM T99685 C6P7JB 136041775 IC50 > 10000 nM T99685 C5CJF7 136041776 IC50 > 10000 nM T99685 C3XIZ8 136041777 IC50 > 10000 nM T99685 C32LKO 136041785 IC50 > 10000 nM T99685 C90ARP 136041787 IC50 > 10000 nM T99685 CG19DI 136041799 IC50 > 10000 nM T99685 CS70RL 136042289 IC50 = 1270 nM T99685 CBHJ83 136042290 IC50 = 2440 nM T99685 C06KNL 136042291 IC50 = 630 nM T99685 CRA3T8 136042292 IC50 = 1050 nM T99685 CKT2U5 136042293 IC50 = 1930 nM T99685 CF3AV4 136042294 IC50 = 780 nM T99685 CZH70G 136042295 IC50 = 2380 nM T99685 CFN2U4 136042296 IC50 = 340 nM T99685 CK28EH 136042297 IC50 = 14100 nM T99685 CKE4R3 136042298 IC50 = 1670 nM T99685 CB0SV5 136042299 IC50 = 178 nM T99685 CQ0DF6 136042300 IC50 = 1040 nM T99685 C89CTO 136066004 IC50 = 32 nM T99685 CLA3C2 136068720 IC50 = 1200 nM T99685 C6ZH2F 136074294 IC50 = 2670 nM T99685 C1SME2 136074295 IC50 = 800 nM T99685 C95LGV 136074296 IC50 = 1940 nM T99685 CAK83X 136074297 IC50 = 6930 nM T99685 CTO47N 136079653 Ki = 2.9 nM T99685 CG1R7B 136087060 IC50 = 770 nM T99685 CC4UM3 136176116 IC50 > 10000 nM T99685 CJRK81 136176117 IC50 > 10000 nM T99685 C63IOS 136176118 IC50 > 10000 nM T99685 C3KW7H 136176119 IC50 > 10000 nM T99685 C69AKQ 136176120 IC50 > 10000 nM T99685 CF17KO 136176121 IC50 > 10000 nM T99685 CU3TE0 136176122 IC50 > 10000 nM T99685 C6C5KB 136176123 IC50 > 10000 nM T99685 C3X5KE 136176124 IC50 > 10000 nM T99685 CA8C5E 136176125 IC50 > 10000 nM T99685 C5OMG2 136176126 IC50 > 10000 nM T99685 CP2YM7 136176127 IC50 > 10000 nM T99685 C8XIJ0 136176128 IC50 > 10000 nM T99685 CUY8N4 136176129 IC50 > 10000 nM T99685 C3J4ME 136176130 IC50 > 10000 nM T99685 CR1NZ2 136176131 IC50 > 10000 nM T99685 C4WG2F 136176132 IC50 > 10000 nM T99685 CJ8EC5 136176139 IC50 > 10000 nM T99685 CHC5U8 136180788 IC50 = 550 nM T99685 C62SVA 136180789 IC50 = 560 nM T99685 C04XFY 136180790 IC50 = 52 nM T99685 CHLD54 136180791 IC50 = 550 nM T99685 CI6HG4 136249373 IC50 = 54 nM T99685 C0GZV9 136254283 IC50 > 10000 nM T99685 C3SJU4 136998793 IC50 = 2200 nM T99685 CH39TP 137453801 Ki = 137 nM T99685 C1EK8U 137453918 Ki = 37.9 nM T99685 CTZA58 137628643 IC50 = 7 nM T99685 C67EFJ 137628684 IC50 = 1.2 nM T99685 CZ5D6V 137631622 IC50 = 39.8 nM T99685 C1NWV2 137631657 IC50 = 222 nM T99685 CMI8E6 137632184 IC50 = 9.9 nM T99685 CN7WS0 137632234 IC50 = 75.8 nM T99685 CX39MO 137632259 IC50 = 31 nM T99685 C7Q2EY 137632337 IC50 = 70 nM T99685 CH8G2L 137632817 IC50 > 2000 nM T99685 CDEX29 137632839 IC50 > 2000 nM T99685 C38JDC 137633109 IC50 = 430 nM T99685 CZ7DR9 137633736 IC50 = 1190 nM T99685 CG73ZQ 137634050 IC50 > 2000 nM T99685 CTIA47 137634248 IC50 = 12 nM T99685 C5Z9FJ 137634261 IC50 = 425 nM T99685 CT40CM 137634322 IC50 > 2000 nM T99685 CCOG91 137634454 IC50 = 632 nM T99685 C6XMW2 137634650 IC50 = 410 nM T99685 CJN3B7 137634657 IC50 = 336 nM T99685 C34MHP 137634951 IC50 = 424 nM T99685 C8Q6WO 137635732 IC50 = 603 nM T99685 C7HBC4 137635822 IC50 = 4 nM T99685 CE4G3W 137635842 IC50 = 15.8 nM T99685 CHZ81K 137635885 IC50 = 104 nM T99685 C3KW5I 137636364 IC50 = 42 nM T99685 C5LHV9 137636943 IC50 = 29 nM T99685 C9UOW1 137637213 IC50 = 301 nM T99685 C5XKI7 137637306 IC50 > 2000 nM T99685 CU0O1W 137637367 IC50 = 422 nM T99685 CRP32A 137637486 IC50 > 2000 nM T99685 CSBY89 137637823 Ki = 660000 nM T99685 CMXV61 137637891 IC50 = 54.3 nM T99685 CO1V2E 137638253 IC50 > 2000 nM T99685 CS78JW 137639139 IC50 = 29000 nM T99685 C04NSI 137639729 IC50 = 26.2 nM T99685 CXZT29 137640462 Ki = 2539 nM T99685 CX1GO6 137641431 IC50 = 40.5 nM T99685 CJI94C 137641546 IC50 = 109 nM T99685 CG0FN1 137641601 IC50 = 167 nM T99685 C47VUG 137642023 IC50 = 54.9 nM T99685 CD2P5V 137642092 IC50 > 2000 nM T99685 CM1OD9 137642750 IC50 = 80 nM T99685 CP4DI5 137643070 IC50 = 330 nM T99685 C3QMK4 137643184 IC50 = 176 nM T99685 C4MVA7 137643536 IC50 > 2000 nM T99685 CUV1A4 137643705 IC50 = 55 nM T99685 C2ABR3 137644061 IC50 = 32 nM T99685 CL96JB 137644395 IC50 = 18.8 nM T99685 CP23NG 137644864 IC50 > 2000 nM T99685 C1O2NP 137645662 IC50 = 23 nM T99685 CI9D4L 137645884 IC50 = 290 nM T99685 CL4J3R 137646575 IC50 > 2000 nM T99685 CQ5T0F 137647241 IC50 = 24 nM T99685 CPMG65 137647250 IC50 = 10 nM T99685 CJ6KD5 137647435 IC50 = 865 nM T99685 C47HXI 137648104 IC50 = 1320 nM T99685 C7B6WC 137648193 IC50 = 4 nM T99685 CR9T0O 137648974 IC50 = 72.3 nM T99685 CK87YT 137649881 IC50 = 612 nM T99685 CECO31 137650069 IC50 = 463 nM T99685 CR6TM0 137650921 IC50 = 53 nM T99685 C7JQC2 137651055 Ki = 185 nM T99685 CI7R1A 137651064 IC50 = 32.9 nM T99685 CMV6K0 137651704 IC50 = 60 nM T99685 CF93QZ 137651837 IC50 = 3 nM T99685 C83KDE 137651894 IC50 = 172 nM T99685 C84TWB 137652545 IC50 = 73 nM T99685 CQMS19 137652991 IC50 > 2000 nM T99685 C5C7OQ 137653159 IC50 = 403 nM T99685 CN1P6C 137653212 IC50 = 201 nM T99685 C2LZE9 137653237 IC50 > 2000 nM T99685 CF4PA2 137654087 IC50 = 8.8 nM T99685 C2EVS5 137654553 IC50 > 2000 nM T99685 CPYL73 137654574 IC50 = 423 nM T99685 C7PF5R 137655359 IC50 = 82.9 nM T99685 C7ON1W 137655398 IC50 = 56 nM T99685 CD7X9E 137655716 IC50 = 3 nM T99685 CM26BD 137655969 IC50 = 14 nM T99685 C4VI2E 137656292 IC50 = 274 nM T99685 C0E8FC 137656416 IC50 = 40.6 nM T99685 CT9U7N 137656570 IC50 = 399 nM T99685 CCZ7P9 137656901 IC50 = 30.8 nM T99685 CA5ZU8 137657493 IC50 > 2000 nM T99685 CL8Z2V 137657573 IC50 = 36.6 nM T99685 CQE1B2 137657755 IC50 = 35 nM T99685 CX0NW5 137658179 IC50 = 3.57 nM T99685 CJ4QT6 137658610 IC50 = 335 nM T99685 C6MB1D 137658961 IC50 = 23.4 nM T99685 CWZ4P7 137659099 IC50 = 225 nM T99685 CT4CL9 137661232 IC50 = 3 nM T99685 CFJ5I9 137661497 IC50 = 427 nM T99685 CN73GX 137661561 IC50 > 2000 nM T99685 C81XWJ 137661590 Ki = 241 nM T99685 CZ25DA 137661970 IC50 = 68 nM T99685 CBS7L6 137662030 IC50 = 270 nM T99685 CA16BS 137662160 Ki = 110000 nM T99685 CA3C4O 138454792 IC50 = 2861 nM T99685 CKDZ26 138504497 IC50 = 5300 nM T99685 CDKR41 139030535 Ki = 8 nM T99685 C1NQ0F 139207772 Ki = 62 nM T99685 C3O5IA 139207773 Ki = 10 nM T99685 CKLH15 139207774 Ki = 4 nM T99685 C26NWP 139486659 Ki = 21.1 nM T99685 CV54CS 141471198 IC50 = 10 nM T99685 C25HYI 141471200 IC50 = 10 nM T99685 CZS03J 141509623 IC50 = 228 nM T99685 C8FZE6 142608579 Ki = 6 nM T99685 CR5GQ3 145949526 IC50 = 3450 nM T99685 C9E6AO 145950785 IC50 = 180 nM T99685 CDOU79 145953070 IC50 = 200 nM T99685 C7DO3I 145953589 IC50 > 10000 nM T99685 CG9F6T 145953725 IC50 = 90 nM T99685 CKQ63F 145955821 IC50 = 330 nM T99685 COC83T 145959468 IC50 = 260 nM T99685 C65YWX 145964882 IC50 > 10000 nM T99685 CHC3T0 145965031 IC50 > 10000 nM T99685 CP92ZF 145965329 IC50 > 10000 nM T99685 C9HXI4 145966620 IC50 > 10000 nM T99685 CQE9M5 145966810 IC50 > 10000 nM T99685 C1EH6C 145967078 IC50 > 10000 nM T99685 CWJ12M 145969155 IC50 > 10000 nM T99685 CGW5S1 145969844 IC50 > 10000 nM T99685 CB8R3A 145970271 IC50 > 10000 nM T99685 C40VIL 145972979 IC50 > 10000 nM T99685 CQBY19 145974023 IC50 > 10000 nM T99685 C4X7CT 145977420 IC50 > 10000 nM T99685 CLA57T 145978300 IC50 > 10000 nM T99685 CZ1T9X 145979969 Ki = 54.3 nM T99685 C03BJC 145980560 Ki = 3.4 nM T99685 CGA83C 145981271 IC50 = 34 nM T99685 CVR1X3 145981509 Ki = 60 nM T99685 CJ1G9L 145981832 Ki = 483 nM T99685 CH6X1R 145983184 Ki = 18.5 nM T99685 CD70WO 145986565 Ki = 435 nM T99685 CH7I9T 145987129 IC50 = 640 nM T99685 C5R6BS 145987142 IC50 = 52 nM T99685 C6D8QS 145987359 Ki = 474 nM T99685 C4BWJ3 145987648 Ki = 551 nM T99685 C9TYO4 145988008 Ki = 74.5 nM T99685 CACF81 145990005 IC50 = 720 nM T99685 C32MJQ 145990827 Ki = 79.9 nM T99685 CSYC93 145991982 Ki = 30 nM T99685 CA0J2B 145992083 Ki = 308 nM T99685 C36RTB 145993509 IC50 = 77.2 nM T99685 C4K0JW 145996540 IC50 = 21 nM T99685 CI85VS 146731761 IC50 = 9380 nM T99685 CLJ63X 147056594 IC50 > 1000 nM T99685 CT5HC9 147206876 IC50 > 1000 nM T99685 C7PI4F 147233226 IC50 = 253 nM T99685 C8TZB7 147371092 IC50 > 1000 nM T99685 CNA3L7 147416694 IC50 > 1000 nM T99685 CNAS83 147431947 IC50 = 48.6 nM T99685 CA21MO 147594782 IC50 > 1000 nM T99685 C05AJN 147697387 IC50 > 1000 nM T99685 CLH9U0 147709166 IC50 > 1000 nM T99685 CUQ8L3 147759183 IC50 = 17.9 nM T99685 CU72AS 147915791 IC50 > 1000 nM T99685 CA3TU9 147919900 IC50 = 267 nM T99685 C2J4TH 147979216 IC50 > 1000 nM T99685 C12CAJ 148039602 IC50 > 1000 nM T99685 CJ8NS7 148093822 IC50 > 1000 nM T99685 CSE50M 148120257 IC50 > 1000 nM T99685 CO0XB2 148191117 IC50 = 873 nM T99685 C5F3IQ 148239318 IC50 = 14.1 nM T99685 C92HBW 148300515 IC50 = 15.3 nM T99685 C74THK 148331443 IC50 > 1000 nM T99685 CZL64V 148493390 IC50 > 1000 nM T99685 CZ1N2T 148551789 IC50 > 1000 nM T99685 CND84O 148558668 IC50 > 1000 nM T99685 CWZ05D 148564044 IC50 = 13.85 nM T99685 CZA3D8 148695436 IC50 > 1000 nM T99685 CHER08 148928697 IC50 > 1000 nM T99685 CI8G9Y 149093021 IC50 = 34.9 nM T99685 CD2LF7 149098844 IC50 > 1000 nM T99685 CNY4Q3 149163842 IC50 = 19.4 nM T99685 COEI42 149296008 IC50 > 1000 nM T99685 CJ80FH 149323347 IC50 > 1000 nM T99685 CN87RZ 149370890 IC50 > 10000 nM T99685 C82BFC 149396423 IC50 > 1000 nM T99685 COMP43 149503998 IC50 > 1000 nM T99685 CK4FJ1 149556361 IC50 = 8120 nM T99685 C2ABX3 152981558 IC50 = 19.8 nM T99685 C7ZU5T 153109924 IC50 = 13.8 nM T99685 C6RFV3 153244706 IC50 > 1000 nM T99685 CU42HJ 153248266 IC50 = 12.6 nM T99685 CJ0EN5 153262665 IC50 > 1000 nM T99685 C8UQL4 153940691 IC50 > 10000 nM T99685 CMZ68Q 153940692 IC50 > 10000 nM T99685 CY2WZ6 155233745 IC50 = 256.8 nM T99685 CDXM69 155249380 IC50 = 7766 nM T99685 CH6V0O 155249545 IC50 = 29.24 nM T99685 C1OVC9 155511557 Ki = 2.5 nM T99685 CG49LC 155512502 IC50 = 3.1 nM T99685 CG9I4X 155512515 IC50 = 7440 nM T99685 CR1Z8A 155512529 IC50 = 5300 nM T99685 C2MD1Q 155513187 IC50 > 10000 nM T99685 CF6CG8 155513897 IC50 > 1000 nM T99685 C17NTI 155514706 Ki = 2200 nM T99685 CEFS61 155515135 IC50 > 10000 nM T99685 CX72DF 155515279 IC50 = 5011.87 nM T99685 CBK3C9 155515384 Ki = 20 nM T99685 CI50FQ 155516321 IC50 > 1000 nM T99685 C8FWK7 155517588 IC50 = 501.19 nM T99685 C5D6YX 155521099 IC50 > 10000 nM T99685 CC1P7U 155521604 IC50 > 1000 nM T99685 CABC57 155522182 Ki = 1700 nM T99685 C5AHS1 155523025 IC50 = 4.3 nM T99685 CZ3FC8 155523374 Ki = 43.1 nM T99685 CZG27I 155523570 IC50 = 676 nM T99685 CG61OL 155524143 IC50 > 1000 nM T99685 CJMD34 155525139 Ki = 190 nM T99685 C9E2PJ 155525385 IC50 = 290.5 nM T99685 C3I9UX 155526450 Ki = 27 nM T99685 CPJ3R6 155526809 Ki = 9.1 nM T99685 C9PF1D 155527778 IC50 = 635 nM T99685 CF2P3Q 155527936 Ki = 1892 nM T99685 CJ3LP5 155528779 Ki = 56 nM T99685 C9OVL5 155528904 Ki = 50 nM T99685 CNA30V 155529246 IC50 > 1000 nM T99685 C9L6OC 155529247 IC50 = 6262 nM T99685 CPH72K 155531472 IC50 > 1000 nM T99685 CA7T0Y 155533911 IC50 > 10000 nM T99685 C68NQP 155536585 Ki = 96 nM T99685 C1Y9MS 155537503 Ki = 2300 nM T99685 CHR8M1 155538990 IC50 = 9120 nM T99685 CE8TV9 155541005 Ki = 40 nM T99685 CN5U9M 155541206 Ki = 34 nM T99685 CYB90C 155542790 Ki = 4000 nM T99685 C8OC2P 155542800 IC50 = 660 nM T99685 CV5L6B 155543139 Ki = 370 nM T99685 CBN29V 155544583 IC50 = 846 nM T99685 C5IVX6 155544961 Ki = 265 nM T99685 CV9OI5 155545359 IC50 = 3.6 nM T99685 CE02BC 155545624 IC50 = 1584.89 nM T99685 CJ1E0T 155547067 Ki = 59.2 nM T99685 CKR36G 155547524 Ki = 39.6 nM T99685 C6JCV4 155548973 Ki = 13 nM T99685 CJWV35 155549094 Ki = 33 nM T99685 C4PEJ5 155549895 IC50 > 10000 nM T99685 CGNF42 155549917 Ki = 76.8 nM T99685 CQ5OD0 155550395 IC50 = 181 nM T99685 CE5DG7 155550972 Ki = 104 nM T99685 CVO9N5 155551369 Ki = 208 nM T99685 CF8D9H 155552080 Ki = 47.8 nM T99685 CJ75BO 155552100 IC50 = 6550 nM T99685 C8L4MZ 155554924 Ki = 85 nM T99685 CCY47Q 155554935 IC50 > 1000 nM T99685 CFW90N 155555562 IC50 = 40 nM T99685 C3BK7O 155556309 Ki = 171 nM T99685 CO4GE3 155557022 Ki = 31 nM T99685 C0FE4G 155557988 IC50 > 10000 nM T99685 C6BAV3 155558720 Ki = 24 nM T99685 CZCO50 155559160 Ki = 300 nM T99685 C7TP0F 155559332 Ki = 60 nM T99685 CVG49I 155560688 IC50 > 10000 nM T99685 C4GXV3 155562151 Ki = 28 nM T99685 C6RV0H 155563416 Ki = 11 nM T99685 CTEB79 155563891 Ki = 31 nM T99685 CC04GI 155564488 IC50 = 31.62 nM T99685 C5SH4P 155565730 Ki = 121 nM T99685 CPA75N 155566172 IC50 = 3.4 nM T99685 C3XMB6 155567232 Ki = 21 nM T99685 C1S8ZB 155568922 IC50 = 3450 nM T99685 CTG81X 155569017 Ki = 177 nM T99685 CUH38L 155569363 IC50 = 8370 nM T99685 CVR2J1 155569607 Ki = 13 nM T99685 D00GQM 25069592 IC50 = 4500 nM T99685 D00JIV 51033720 Ki = 1440 nM T99685 D02TCF 44576240 IC50 = 5 nM T99685 D02TSN 46244454 IC50 = 38 nM T99685 D03EHM 24905142 IC50 = 10 nM T99685 D03QQH 16760391 IC50 > 100000 nM T99685 D05BPX 9901372 IC50 = 49 nM T99685 D05USL 5278396 IC50 = 5580 nM T99685 D06HVH 54613583 IC50 > 9100 nM T99685 D07JKB 135955185 IC50 = 2500 nM T99685 D07PMP 44187953 IC50 = 1.7 nM T99685 D09FBN 135955186 IC50 = 450 nM T99685 D0AH8Q 25074311 IC50 = 2800 nM T99685 D0F1SI 25074312 IC50 = 3900 nM T99685 D0H0HR 49836027 IC50 = 4.32 nM T99685 D0H2CM 135565635 IC50 = 8 nM T99685 D0R0TW 11964036 IC50 = 10000 nM T99685 D0T0BY 10039361 IC50 = 5300 nM T99685 D0TC5H 16049458 IC50 = 1650 nM T99685 D0U8GR 44576241 IC50 = 10 nM T99685 D0W1ST 9860529 IC50 = 6400 nM T99685 D0W8XH 9884685 IC50 = 8.8 nM T99685 D0X7TB 10017389 IC50 = 4800 nM T99685 D0Y1DR 46225260 IC50 = 150 nM T99685 D0Y3OO 11327430 IC50 = 1700 nM T70019 D03RTS 2662 IC50 > 40000 nM T70019 D06GDY 43815 IC50 = 7000 nM T70019 D09XZB 123631 IC50 = 9700 nM T70019 D0E6XR 3062316 IC50 = 11500 nM T70019 D0J4JM 5770 IC50 = 7000 nM T70019 D0T0KA 4474 IC50 = 22800 nM T70019 CE2OY6 92783 IC50 = 15000 nM T70019 CUE30K 3863543 IC50 = 6800 nM T70019 CW2NG6 4130365 IC50 = 5800 nM T70019 CLE82K 4180540 IC50 = 17000 nM T70019 CS5K7W 5729232 IC50 = 29100 nM T70019 C1ZPG8 5930244 IC50 = 26500 nM T70019 C8TD9Z 6280084 IC50 = 15000 nM T70019 C4I5DA 7946175 IC50 = 24300 nM T70019 CZ1L7K 10826895 IC50 = 13400 nM T70019 CX75AR 24014552 IC50 = 22500 nM T70019 C6WH3J 53316933 IC50 = 8900 nM T70019 CSY82V 53322217 IC50 = 7300 nM T70019 CRW6I8 57384550 IC50 = 10000 nM T70019 CL27ZC 60141344 IC50 = 18000 nM T70019 C8PDI5 71451413 IC50 = 7700 nM T70019 CABI32 71453222 IC50 = 18100 nM T70019 CT48MG 71454950 IC50 = 9000 nM T70019 CAJ7O6 71456744 IC50 = 28400 nM T70019 C4OVL6 71456745 IC50 = 16900 nM T70019 CD8I5Q 71734010 IC50 = 9900 nM T70019 CK0HT4 71734012 IC50 = 13300 nM T70019 CJS41D 71734013 IC50 = 7500 nM T70019 CMO94A 71734014 IC50 = 8000 nM T70019 C0AP4O 71734015 IC50 = 14800 nM T70019 CN4W1E 71734109 IC50 = 8300 nM T70019 C4FI7N 71734110 IC50 = 3900 nM T70019 CJQC60 71734112 IC50 = 10700 nM T70019 CLPC48 71734113 IC50 = 9300 nM T70019 CQ6Z3H 71734114 IC50 = 6400 nM T70019 CLG31J 71734202 IC50 = 8300 nM T70019 CLE2V0 71734203 IC50 = 9700 nM T70019 C4IT0S 71734204 IC50 = 3800 nM T70019 CF0L6N 71734299 IC50 = 9200 nM T70019 CNZ08Y 71734302 IC50 = 8500 nM T70019 CAI92Q 71734303 IC50 = 9300 nM T70019 C6ITD3 127029910 IC50 = 10600 nM T70019 C4SP8G 127029911 IC50 = 11900 nM T70019 CF3Q0S 127029912 IC50 = 12500 nM T70019 CPN69V 127030216 IC50 = 6600 nM T70019 CRW4D6 127030501 IC50 = 17100 nM T70019 CY39GC 127030512 IC50 = 13700 nM T70019 CI7Y4M 127030513 IC50 = 4800 nM T70019 C0NOA5 127030514 IC50 = 6100 nM T70019 CAZS58 127030515 IC50 = 6700 nM T70019 CAE18G 127031175 IC50 = 11600 nM T70019 C90UTN 127031176 IC50 = 16800 nM T70019 C3R2EJ 127032061 IC50 = 10400 nM T70019 CKR1D6 127032062 IC50 = 5100 nM T70019 CZF2B4 127032333 IC50 = 14200 nM T70019 COLB92 127032334 IC50 = 14100 nM T70019 C35AGS 127032335 IC50 = 6300 nM T70019 C3DER4 127032336 IC50 = 4400 nM T70019 C2VSI0 127032337 IC50 = 6500 nM T70019 CU9F1Y 127032338 IC50 = 6100 nM T70019 CTW02C 127032933 IC50 = 12500 nM T70019 C7QB6T 127032936 IC50 = 15500 nM T70019 C9QCS3 127033275 IC50 = 5000 nM T70019 CJOR74 127033276 IC50 = 7300 nM T70019 C6D4KG 127033277 IC50 = 7100 nM T70019 C3CR1G 127033278 IC50 = 4800 nM T70019 C3GDY4 127033317 IC50 = 6700 nM T70019 CZM1X2 127033556 IC50 = 6100 nM T70019 CW63OP 127033557 IC50 = 8700 nM T70019 CP0EB9 127034433 IC50 = 10100 nM T70019 CMV50U 127034434 IC50 = 6000 nM T70019 C85IFB 134141646 IC50 = 1800 nM T70019 CY8EV3 134144287 IC50 = 2020 nM T70019 CILP41 134144373 IC50 = 4930 nM T70019 CW1R3V 134146455 IC50 = 19900 nM T70019 CNZT90 134148138 IC50 = 3830 nM T70019 CR5LF1 137640351 IC50 = 2000 nM T70019 CJ8QR6 145949258 IC50 = 4700 nM T70019 C3SIY5 145950318 IC50 = 1800 nM T70019 CRYX41 145950443 IC50 = 1600 nM T70019 CRT5W7 145950615 IC50 = 10600 nM T70019 CTO8M9 145950651 IC50 = 4700 nM T70019 C4HF1J 145950697 IC50 = 1100 nM T70019 CFL06Z 145951132 IC50 = 9900 nM T70019 C6FQT3 145951725 IC50 = 4400 nM T70019 CFV4W5 145951762 IC50 = 3300 nM T70019 C9E3UY 145951822 IC50 = 5500 nM T70019 C4TEI7 145952799 IC50 = 4600 nM T70019 C80YWC 145953257 IC50 = 3800 nM T70019 C2QZA9 145953508 IC50 = 3800 nM T70019 CW24KI 145953601 IC50 = 4900 nM T70019 CUH18V 145954056 IC50 = 5200 nM T70019 C0AIN2 145954370 IC50 = 5000 nM T70019 CU0BW3 145954413 IC50 = 11900 nM T70019 C62SDY 145955072 IC50 = 9400 nM T70019 CYD7V3 145955275 IC50 = 7300 nM T70019 CZK19B 145955384 IC50 = 5800 nM T70019 CNUR70 145956269 IC50 = 8100 nM T70019 C9OPW0 145957472 IC50 = 4000 nM T70019 CQ79DH 145957562 IC50 = 3300 nM T70019 C65MRZ 145957810 IC50 = 3900 nM T70019 C3X7HJ 145958704 IC50 = 4200 nM T70019 C9IRA2 145958815 IC50 = 4700 nM T70019 C69GZE 145958958 IC50 = 4100 nM T70019 C39UTB 145959055 IC50 = 7200 nM T70019 C16WTI 145959243 IC50 = 2800 nM T70019 CH8VK6 145959665 IC50 = 19100 nM T70019 C8FQ7L 145960310 IC50 = 13700 nM T70019 C8G9YV 145961007 IC50 = 8800 nM T70019 CF89DI 145972663 IC50 = 4300 nM T70019 CR57XJ 145972709 IC50 = 2200 nM T70019 CJ81VR 145973585 IC50 = 4100 nM T70019 C8NO7Q 145974098 IC50 = 15600 nM T12005 D02UOE 160142 Ki = 21500 nM T12005 CG9P4V 70871 IC50 = 25000 nM T12005 C7KJ3B 114917 Ki = 13700 nM T12005 C5X1YU 160254 IC50 = 800 nM T12005 C4IRY2 164676 IC50 = 1600 nM T12005 CHS3V9 318797 IC50 = 18000 nM T12005 CK5V1Q 515954 Ki = 71000 nM T12005 C8PNR0 515962 IC50 = 12500 nM T12005 CX5O0F 515964 Ki = 120 nM T12005 CHG4X9 1342108 IC50 = 500000 nM T12005 C1L3ZF 2726174 IC50 = 13000 nM T12005 C3WV6Q 2726176 IC50 = 13000 nM T12005 C8NCQ7 2742278 IC50 = 10000 nM T12005 C0O4DB 2745617 IC50 = 15000 nM T12005 C9V7QZ 2745640 IC50 = 15000 nM T12005 CG8K7V 2745653 IC50 = 15000 nM T12005 CGED72 2774667 IC50 = 15000 nM T12005 CFV57C 2774892 IC50 = 900 nM T12005 C46ZTR 2775844 IC50 = 16000 nM T12005 CUIA69 2797358 IC50 = 12000 nM T12005 CT86VO 2799606 IC50 = 300 nM T12005 CH8X5M 2799800 IC50 = 32000 nM T12005 CGCX02 2799801 IC50 = 16000 nM T12005 C0XG4Q 2800273 IC50 = 95 nM T12005 C7U6ND 2810524 IC50 = 250000 nM T12005 C3T8PB 2819040 IC50 = 6000 nM T12005 CUA3V8 2820775 IC50 = 16000 nM T12005 CXF53O 2820912 IC50 = 11000 nM T12005 C0ZSF7 2821293 IC50 = 10000 nM T12005 C4OQ7Y 2822496 IC50 = 3000 nM T12005 CXYA78 2823615 IC50 = 400000 nM T12005 CQ30AR 2918713 IC50 = 300000 nM T12005 CPXI87 3776668 IC50 = 5000 nM T12005 CE68DQ 4270495 IC50 = 16000 nM T12005 CJ7PV5 4305683 IC50 = 20000 nM T12005 CG9V1A 4398304 IC50 = 18000 nM T12005 COIX12 6476897 Ki > 10000 nM T12005 CJ8YG9 6478229 Ki = 2260 nM T12005 C8VJ3P 7230550 IC50 = 60 nM T12005 C8K2NO 10062715 IC50 = 70000 nM T12005 CJP85S 10642441 Ki = 50000 nM T12005 CJ82DN 10645393 Ki = 1096.48 nM T12005 C1JAC5 11425923 IC50 = 1200 nM T12005 C4UVG8 11444522 Ki = 660 nM T12005 CGAF41 11456186 Ki = 53 nM T12005 CH6JQ1 11515424 Ki = 66000 nM T12005 C01USX 11630144 Ki = 19000 nM T12005 C6GN2F 11642725 IC50 = 45000 nM T12005 C5UJH3 11644322 Ki = 25000 nM T12005 CSP38Q 11667869 IC50 = 980 nM T12005 CGJO74 11786957 Ki = 58 nM T12005 CNK98D 11796320 IC50 = 950 nM T12005 CB42PF 14610613 IC50 = 9200 nM T12005 C68KOL 16203681 IC50 = 50 nM T12005 CF90EY 16203796 IC50 = 270 nM T12005 C58WAX 16203797 IC50 = 63 nM T12005 CLY71W 16204318 IC50 = 170 nM T12005 CZE4V3 16204322 IC50 = 65 nM T12005 CJ6Y0I 16204324 IC50 = 340 nM T12005 C5QZB4 44398002 IC50 = 9400 nM T12005 CGW7K3 44398055 IC50 = 13110 nM T12005 CIM7Q2 44398160 IC50 = 7200 nM T12005 C7FEW1 44398167 IC50 = 13500 nM T12005 CTDN81 44398207 IC50 = 4820 nM T12005 C8RQ4W 44398231 IC50 = 23500 nM T12005 C4J1GY 44398343 IC50 = 2000 nM T12005 CY52ZS 44398344 IC50 = 11200 nM T12005 C02BZJ 44398436 IC50 = 17500 nM T12005 C1A9KO 44398546 IC50 = 12570 nM T12005 C2YZQ1 44415162 IC50 = 15000 nM T12005 CC6NL2 44415172 IC50 = 18000 nM T12005 CV0IX7 44415173 IC50 = 40000 nM T12005 CGSD17 135408428 IC50 = 100000 nM T12005 CRMN90 135411083 IC50 = 40000 nM T12005 C7Q2EG 135411084 IC50 = 60000 nM T12005 C13ZPV 135411086 IC50 = 200000 nM T12005 C43ECP 135411087 IC50 = 200000 nM T12005 CN5W1R 135411089 IC50 = 300000 nM T12005 C0V7GK 135411090 IC50 = 350000 nM T12005 C72ZIQ 135411091 IC50 > 1000000 nM T12005 C8T3AC 135419065 IC50 = 200000 nM T12005 CMNA95 135427623 IC50 = 300000 nM T12005 CA0IU9 135442547 IC50 = 30000 nM T12005 CZMO07 136106200 IC50 = 60000 nM T56121 D0E3TC 44259 IC50 = 1830 nM T56121 D04FHB 6918852 Ki > 5000 nM T56121 D0T3ME 156422 IC50 = 9400 nM T56121 C2TC1L 9910609 IC50 = 1090 nM T56121 C64IGY 11448608 Ki > 5000 nM T56121 CG92CF 46175112 IC50 = 1000 nM T56121 CZW06V 46175113 IC50 = 79 nM T56121 CFN9J6 46175114 IC50 = 228 nM T56121 CJ24EK 46175116 IC50 = 87 nM T56121 C25NWI 46882439 IC50 = 20000 nM T56121 C9WKA2 46882442 IC50 = 20000 nM T56121 CB6OR2 46882444 IC50 = 20000 nM T56121 COTP05 46882506 IC50 = 20000 nM T56121 C3QN6Y 46882510 IC50 = 20000 nM T56121 CDO70W 46882511 IC50 = 20000 nM T56121 CQNF38 46882512 IC50 = 15000 nM T56121 C3DBI8 46882570 IC50 = 260 nM T56121 CX9J4F 46882571 IC50 = 15000 nM T56121 CQR1B0 46882573 IC50 = 20000 nM T56121 CIX89V 46882574 IC50 = 2000 nM T56121 CU0H5K 46882575 IC50 = 20000 nM T56121 C0H3ZY 46882576 IC50 = 190 nM T56121 CJB8C4 46882615 IC50 = 66 nM T56121 C1JFW0 46882616 IC50 = 77 nM T56121 CGY04I 46882617 IC50 = 200 nM T56121 CE05QG 46882618 IC50 = 240 nM T56121 C0FK7D 46882619 IC50 = 63 nM T56121 CXLI61 46882659 IC50 = 20000 nM T56121 C3A9XD 46882662 IC50 = 20000 nM T56121 CI5WT8 46882663 IC50 = 20000 nM T56121 CKF1I5 46882704 IC50 = 15000 nM T56121 C6C9HP 46882706 IC50 = 460 nM T56121 CS9A3L 46882707 IC50 = 60 nM T56121 CX3H2C 46882742 IC50 = 20000 nM T56121 CY9HN3 46882743 IC50 = 20000 nM T56121 C2GB6O 46882745 IC50 = 173 nM T56121 C8NA4L 53384644 IC50 > 30000 nM T56121 CE1A9V 57394653 IC50 = 350 nM T56121 CV63UL 67240318 IC50 > 10000 nM T56121 C9WGB8 127035904 IC50 = 3900 nM T56121 C2KFH7 135398497 Ki > 2000 nM T56121 CS4OW8 135400873 Ki > 2000 nM T56121 CFAD48 135611170 Ki > 2000 nM T56121 C2MD1Q 155513187 IC50 > 10000 nM T56121 D05FXD 44478401 IC50 = 15 nM T56121 D09XIL 11396738 IC50 = 1250 nM T56121 D0X8BU 71718651 IC50 = 4400 nM T08391 D03ZBT 11626560 IC50 = 27 nM T08391 D04LKS 25126798 IC50 = 0.056 nM T08391 D04LVK 57379345 IC50 = 610 nM T08391 D07POC 176870 IC50 = 4000 nM T08391 D0E7PQ 5311 IC50 > 10000 nM T08391 D0EG1I 9926791 IC50 = 0.6 nM T08391 D0J9ZR 4477 IC50 = 10000 nM T08391 D0Y7IC 44205240 IC50 = 5.7 nM T08391 D00DRL 44137946 IC50 = 230 nM T08391 D00RYA 16750271 IC50 = 46 nM T08391 D02TUL 118115473 IC50 > 10000 nM T08391 D03LWG 53235510 IC50 = 2882 nM T08391 D04QWQ 59422203 Ki = 13 nM T08391 D05PCM 78323835 IC50 = 803 nM T08391 D05PZB 135398495 IC50 = 1 nM T08391 D06DMQ 59472121 Ki = 150 nM T08391 D06EIC 57928403 IC50 = 5 nM T08391 D07EHV 44814409 IC50 > 10000 nM T08391 D07HPJ 11476171 IC50 > 10000 nM T08391 D07JAG 58557659 IC50 = 120 nM T08391 D08DHN 67286591 Ki > 4000 nM T08391 D08HOM 46207586 IC50 > 10000 nM T08391 D0BI3N 44595079 IC50 = 6 nM T08391 D0D5ZJ 25062766 IC50 = 18 nM T08391 D0D8KQ 25127112 IC50 = 28 nM T08391 D0DK5X 135567296 IC50 = 23.1 nM T08391 D0DK8X 50922691 IC50 = 80 nM T08391 D0E3TC 44259 IC50 = 0.189 nM T08391 D0G8BM 16722836 IC50 = 3 nM T08391 D0G9AW 59473233 EC50 = 453 nM T08391 D0H2HZ 60194098 IC50 = 10000 nM T08391 D0MP0X 16659841 IC50 < 3 nM T08391 D0O0LS 25141092 IC50 = 40 nM T08391 D0O6WV 24794418 IC50 > 2000 nM T08391 D0P0KN 16739650 IC50 = 73 nM T08391 D0P1CV 46191454 IC50 > 10000 nM T08391 D0PN8H 46216796 IC50 = 1 nM T08391 D0R9IU 44462758 IC50 = 1750 nM T08391 D0S1XX 134821691 IC50 > 10000 nM T08391 D0S6TK 11213558 IC50 = 6 nM T08391 D0SG7B 49831257 IC50 = 2400 nM T08391 D03BNU 59604787 IC50 > 3500 nM T08391 D05PDI 46224913 Ki = 1 nM T08391 D0Y2PO 71770709 IC50 = 16600 nM T08391 D08DBE 10344820 Ki = 130 nM T08391 D0GZ7B 5328779 IC50 > 10000 nM T08391 D0T3ME 156422 IC50 > 30000 nM T08391 CBPM40 4878 IC50 > 50000000 nM T08391 CU68FI 78893 Ki = 3200 nM T08391 C6ZB4U 790291 Ki = 3000 nM T08391 CZJB27 817910 IC50 = 40900 nM T08391 CGQM48 869412 Ki = 1700 nM T08391 C0XL5P 951379 Ki > 3500 nM T08391 C7ZUW6 1246120 Ki = 2800 nM T08391 CI1B7L 1247281 Ki = 3200 nM T08391 CP6BI3 1481965 IC50 = 13000 nM T08391 C19-AUG 1927544 IC50 = 15000 nM T08391 CY35GB 2241431 IC50 = 6000 nM T08391 C4J8HV 2389948 IC50 = 13800 nM T08391 CWCH42 2786631 IC50 = 131000 nM T08391 C3F0GS 3120536 Ki = 1200 nM T08391 CD67OL 4250390 Ki > 3500 nM T08391 C6SNL5 4393251 Ki > 3500 nM T08391 CG9RD4 4448318 IC50 = 453 nM T08391 CK6L3O 5121684 Ki = 1700 nM T08391 CX01FS 5473838 IC50 = 60 nM T08391 CGYE97 6419765 IC50 = 61 nM T08391 C2OL7K 9796455 IC50 > 50000 nM T08391 CYA76E 9798589 IC50 > 100000 nM T08391 CQ89SE 9947841 IC50 = 600 nM T08391 CO70CQ 10107882 IC50 = 58 nM T08391 C7SFI1 10296883 IC50 > 10000 nM T08391 C7HBP6 10429593 IC50 > 10000 nM T08391 CBOP58 11293798 Ki > 10000 nM T08391 C26BZX 11362471 Ki > 10000 nM T08391 CWXB93 11397177 Ki > 10000 nM T08391 CT3VP7 11398307 IC50 = 25000000 nM T08391 CK83CN 11416425 IC50 = 40 nM T08391 CTG83F 11539329 Ki > 1500 nM T08391 CI0X1C 11567474 IC50 = 688 nM T08391 CMIL86 11590363 Ki > 1500 nM T08391 CDIW70 11597571 IC50 = 92 nM T08391 C0O3HT 11601868 IC50 = 790 nM T08391 CV8EU0 11612136 IC50 = 65 nM T08391 C9ZD2E 11626406 IC50 = 4891 nM T08391 CSM62L 11626920 IC50 = 29000 nM T08391 C9T6SC 11640926 Ki > 1500 nM T08391 CXG5W8 11646595 IC50 = 3 nM T08391 C5LHC6 11658542 IC50 = 145300 nM T08391 CP3U0W 11684933 IC50 > 8333 nM T08391 CU0E8O 11690457 Ki = 400 nM T08391 CB0AP2 11705863 Ki = 4400 nM T08391 CS36BH 11843159 IC50 = 240 nM T08391 C61TIL 11844913 IC50 = 333 nM T08391 C9JT4S 11847343 IC50 = 1721 nM T08391 CHR92S 11858109 IC50 = 3400 nM T08391 CNYB84 11951225 IC50 = 83 nM T08391 CASK85 11957393 IC50 = 5.9 nM T08391 C58YUH 11993785 IC50 = 30 nM T08391 CW53JC 11998038 Ki = 13 nM T08391 C0Y7MG 12083227 IC50 = 45000 nM T08391 C75SGK 12997800 IC50 = 3 nM T08391 CM9JA0 12997805 IC50 = 0.2 nM T08391 C0DUA7 15953425 IC50 = 4.4 nM T08391 C3JWA6 15953427 IC50 = 3.6 nM T08391 CWZM24 15953526 IC50 = 18 nM T08391 CFPW41 16007116 Ki > 1400 nM T08391 C12TIL 16058762 IC50 = 3 nM T08391 C1WJ2D 16070041 IC50 = 100 nM T08391 COIK65 16070059 IC50 = 150 nM T08391 C1U8XW 16109036 IC50 = 550 nM T08391 CGC34R 16118737 IC50 > 1030 nM T08391 CT8WS0 16126645 IC50 = 124 nM T08391 C5VPH9 16129448 IC50 = 57 nM T08391 CM32VW 16659676 IC50 = 4 nM T08391 CO3L1Q 16659677 IC50 = 10 nM T08391 CL38VY 16659680 IC50 < 3 nM T08391 C5LP4O 16659681 IC50 = 3 nM T08391 C0ECA7 16659682 IC50 = 4 nM T08391 CXYV28 16659836 IC50 < 3 nM T08391 CDTG08 16659837 IC50 < 3 nM T08391 C91SVD 16659838 IC50 < 3 nM T08391 CC10IO 16662069 IC50 = 4 nM T08391 CD1NT2 16662070 IC50 < 3 nM T08391 C19KHB 16664854 IC50 = 209 nM T08391 CO7E8C 16678106 IC50 = 104 nM T08391 C4TC3X 16722832 IC50 = 6 nM T08391 CY1E2N 16723801 IC50 = 133600 nM T08391 C4Q2TN 16739431 IC50 = 210 nM T08391 CWI96A 16739432 IC50 = 62 nM T08391 CSE35D 16739464 IC50 = 820 nM T08391 C20OFQ 16739508 IC50 = 330 nM T08391 CNFX02 16739511 IC50 = 82 nM T08391 C3AGL1 16739512 IC50 = 150 nM T08391 C0JTZ9 16739677 IC50 = 1700 nM T08391 C4IX1K 16739678 IC50 = 510 nM T08391 COZ7A1 16739706 IC50 = 1500 nM T08391 C0HB9T 16739709 IC50 = 1500 nM T08391 C0U8DY 16739710 IC50 = 120 nM T08391 COC6L0 16739741 IC50 > 10000 nM T08391 C1Z8WO 16739742 IC50 = 280 nM T08391 CPT2G0 16739743 IC50 > 10000 nM T08391 CPC5Q9 16739745 IC50 > 10000 nM T08391 CLY96T 16739777 IC50 = 90 nM T08391 C0TMW8 16739778 IC50 = 180 nM T08391 C1MAE7 16739807 IC50 > 10000 nM T08391 C9H8XT 16739808 IC50 > 10000 nM T08391 CC5UB1 16739809 IC50 = 3300 nM T08391 CQ43TS 16739810 IC50 = 48 nM T08391 CJCN32 16739811 IC50 > 10000 nM T08391 CDK6A4 16739812 IC50 = 120 nM T08391 CE0I5O 16739835 IC50 = 160 nM T08391 C4C7DF 16739839 IC50 = 49 nM T08391 C20BPQ 16739840 IC50 = 56 nM T08391 CE1XT6 16739866 IC50 = 1350 nM T08391 C8JBR9 16739867 IC50 = 220 nM T08391 C1VG0U 16739870 IC50 = 62 nM T08391 C2Z4DB 16739901 IC50 = 110 nM T08391 C1UFH7 16739902 IC50 = 220 nM T08391 C7DFM1 16739903 IC50 = 1600 nM T08391 CHX86I 16739904 IC50 = 720 nM T08391 CCP56J 16739905 IC50 = 90 nM T08391 CP9C6B 16739918 IC50 = 100 nM T08391 CJB7M2 16739919 IC50 = 50 nM T08391 C2WNB4 16739920 IC50 = 50 nM T08391 CQ64XI 16739921 IC50 = 170 nM T08391 C9MT8U 16739933 IC50 = 140 nM T08391 CM3UF8 16739935 IC50 = 1100 nM T08391 CFEP56 16739948 IC50 = 260 nM T08391 CKE6V9 16739949 IC50 = 230 nM T08391 C23KZR 16739951 IC50 > 10000 nM T08391 C6GJ5Q 16739952 IC50 = 44 nM T08391 CFRU87 16739965 IC50 = 150 nM T08391 C9OQ1G 16750272 IC50 = 220 nM T08391 CW2SY5 16750291 IC50 = 7.3 nM T08391 CIX7U2 16750304 IC50 = 67 nM T08391 C6A3XS 16750306 IC50 = 17 nM T08391 CB2TK1 16750327 IC50 = 110 nM T08391 CH4O1C 16750328 IC50 = 290 nM T08391 C90MJD 16750331 IC50 = 930 nM T08391 C9MNP2 17549086 IC50 = 8900 nM T08391 CL9BQ6 17748275 IC50 = 1746 nM T08391 C6UAZ0 20820292 IC50 >= 10000 nM T08391 CE7K3W 23532567 IC50 > 10000 nM T08391 C1O6ME 23581858 IC50 = 210 nM T08391 C9WRS3 23581859 IC50 = 52 nM T08391 CYH2Z8 23582563 IC50 = 210 nM T08391 CWEC02 23582564 IC50 = 49 nM T08391 CRO1A2 23582565 IC50 = 230 nM T08391 CD7M2U 23582566 IC50 = 230 nM T08391 CZF6W3 23582567 IC50 = 68 nM T08391 CXZ87O 23582568 IC50 = 190 nM T08391 C6O5JX 23582570 IC50 = 17 nM T08391 CHS9L8 23582639 IC50 = 74 nM T08391 C53OJF 23582642 IC50 = 83 nM T08391 CM9A4G 23582643 IC50 = 51 nM T08391 CBC4Y7 23582701 IC50 = 18 nM T08391 CUY98W 23585560 IC50 = 19 nM T08391 CD0R9O 24699546 Ki = 3200 nM T08391 C7YG1N 24759534 IC50 = 2400 nM T08391 CAJ4T2 24762205 IC50 > 10000 nM T08391 CQNP54 24764449 IC50 = 25000 nM T08391 CFS2M7 24798487 Ki = 59.7 nM T08391 CLBP72 24798571 IC50 = 138 nM T08391 CX1U4S 24800423 IC50 = 15 nM T08391 C4T0DG 24800602 IC50 = 840 nM T08391 CH3ZG7 24800604 IC50 = 440 nM T08391 CBA02Y 24800776 IC50 = 8 nM T08391 C3UFG1 24801129 IC50 = 5 nM T08391 CVR8S1 24801650 IC50 = 110 nM T08391 CV5RP8 24809765 IC50 = 695 nM T08391 C29ANE 24809801 IC50 = 615 nM T08391 C59FKG 24860777 IC50 = 900 nM T08391 CL0O9E 24877325 IC50 = 12.6 nM T08391 CY0P4X 24877326 IC50 = 3.6 nM T08391 C7R4YV 24877438 IC50 = 6.9 nM T08391 C5G4BY 24877439 IC50 = 4.2 nM T08391 C5NXH3 24877440 IC50 = 6.5 nM T08391 CJ4Z0K 24877791 IC50 = 5.1 nM T08391 CQUH61 24877795 IC50 = 11.1 nM T08391 CO5RV2 24878018 IC50 = 4.4 nM T08391 CH3Q1D 24878130 IC50 = 39.6 nM T08391 CFK2B9 24882503 IC50 > 10000 nM T08391 CWV98O 24899557 IC50 = 1600 nM T08391 CLZ23U 24951610 IC50 = 21000 nM T08391 C5S7XA 24958852 IC50 = 41 nM T08391 CJ68PR 24958855 IC50 = 100 nM T08391 CZ18IU 24963047 IC50 = 78 nM T08391 CS3Q8B 24995659 Ki > 4000 nM T08391 CT07ZW 25030805 IC50 = 3 nM T08391 CHLC27 25052652 IC50 = 25 nM T08391 C7W6FX 25059112 IC50 = 8 nM T08391 CD0T4Z 25059626 IC50 = 116 nM T08391 CD4TJ7 25059891 IC50 = 374 nM T08391 CE9N8F 25060146 IC50 = 10 nM T08391 C3Y7SB 25060677 IC50 = 186 nM T08391 CWZH04 25060922 IC50 = 41 nM T08391 C7VPB2 25060927 IC50 = 30 nM T08391 C25NMK 25061435 IC50 = 163 nM T08391 CLH91O 25061438 IC50 = 326 nM T08391 CF3Z0Q 25061949 IC50 = 113 nM T08391 CF3QE4 25061950 IC50 = 549 nM T08391 C2BEQ3 25062226 IC50 = 132 nM T08391 CSVH95 25062228 IC50 = 303 nM T08391 C9KY0J 25062498 IC50 = 65 nM T08391 CG4U2Y 25062765 IC50 = 545 nM T08391 C2FI3E 25062767 IC50 = 533 nM T08391 CVI87D 25063021 IC50 = 52 nM T08391 C4JO2C 25063023 IC50 = 298 nM T08391 C3VIR1 25063025 IC50 = 166 nM T08391 C2KY1G 25094210 IC50 > 10000 nM T08391 C2H4VG 25096016 IC50 = 1 nM T08391 C9YVJ0 25096019 IC50 = 75 nM T08391 C8DTP7 25096020 IC50 = 27 nM T08391 CQA4V6 25096276 IC50 = 53 nM T08391 C40GWA 25096277 IC50 = 1115 nM T08391 CF7TP1 25096279 IC50 = 750 nM T08391 C2V4IM 25096280 IC50 = 100 nM T08391 C05XPV 25096532 IC50 = 4100 nM T08391 CV8PC6 25097027 IC50 = 540 nM T08391 CUB4W5 25102935 IC50 = 5 nM T08391 CM0O7N 25102936 IC50 < 3 nM T08391 C3PKV4 25102938 IC50 < 3 nM T08391 CNQ07G 25103042 IC50 = 6 nM T08391 C09PMH 25103279 IC50 = 3 nM T08391 C1V7QM 25103281 IC50 = 4 nM T08391 COP15B 25103284 IC50 = 17 nM T08391 CP8GU7 25104502 IC50 = 5 nM T08391 C7EK6V 25104503 IC50 = 6 nM T08391 C63ADF 25104611 IC50 = 37 nM T08391 CPM6S0 25104740 IC50 < 3 nM T08391 CJW1T2 25104741 IC50 = 3 nM T08391 CON1U6 25110598 IC50 = 7.5 nM T08391 C0JYA9 25123154 IC50 = 72 nM T08391 C56JVD 25123155 IC50 = 13 nM T08391 CZM6Q2 25123472 IC50 = 5.1 nM T08391 C3IA7V 25123474 IC50 = 120 nM T08391 C6V4NB 25123475 IC50 = 20 nM T08391 C0KOU6 25123487 IC50 = 34 nM T08391 CFK89A 25123806 IC50 = 14 nM T08391 C3RMN9 25123807 IC50 = 20 nM T08391 C5GO3T 25123808 IC50 = 195 nM T08391 C0W8IC 25124143 IC50 = 20 nM T08391 C61WOA 25127137 IC50 = 65 nM T08391 CTPV83 25127138 IC50 = 270 nM T08391 C8ASE3 25127139 IC50 = 398 nM T08391 CY32NR 25127140 IC50 = 178 nM T08391 C2K6UF 25127142 IC50 = 161 nM T08391 C6O4ES 25127144 IC50 = 227 nM T08391 CVQT51 25127461 IC50 = 146 nM T08391 C3UM5H 25127784 IC50 = 891 nM T08391 CF2W8C 25127785 IC50 = 16 nM T08391 C4WFL0 25128110 IC50 = 42 nM T08391 CWD72X 25128951 Ki = 1.6 nM T08391 CM86LX 25128955 Ki = 4200 nM T08391 C56TUK 25128956 Ki = 71 nM T08391 CXJ02U 25129311 Ki = 3100 nM T08391 CHD16N 25129655 Ki = 2 nM T08391 CS1FT7 25130358 Ki = 2400 nM T08391 C6G4DB 25130691 Ki = 2400 nM T08391 C6PAD3 25130693 Ki = 4 nM T08391 C6PXJ0 25130695 Ki = 1500 nM T08391 C9N6KS 25131017 Ki = 200 nM T08391 CND06Y 25131018 Ki = 130 nM T08391 C7GR4S 25131021 Ki = 1300 nM T08391 CF7PV8 25131681 Ki = 56 nM T08391 CFZ23Q 25132021 Ki = 280 nM T08391 CM9O4G 25132023 Ki = 210 nM T08391 C7AY6L 25132025 Ki = 1000 nM T08391 CE20BM 25132384 Ki = 1100 nM T08391 CZO81Q 25132387 Ki = 2000 nM T08391 CXI03Y 25132388 Ki = 3400 nM T08391 C9OCM7 25132389 Ki = 1700 nM T08391 C2NXD1 25132390 Ki = 750 nM T08391 CAL6Y5 25132729 Ki = 490 nM T08391 CE52HX 25132730 Ki = 2900 nM T08391 CS7TM1 25132733 Ki = 210 nM T08391 C9DYQ1 25133399 Ki = 220 nM T08391 COV8Z0 25143021 IC50 > 10000 nM T08391 C6BWZ8 25145145 IC50 > 100 nM T08391 C78YWA 25145716 IC50 > 500 nM T08391 CI0E2L 25154395 IC50 = 18 nM T08391 CL1W5D 25154436 IC50 = 14 nM T08391 CB21XV 25164469 Ki = 91 nM T08391 CUX83H 25164675 Ki = 351 nM T08391 C1H7BF 25164677 Ki = 482 nM T08391 C6SD2A 25165081 Ki > 1453 nM T08391 C67TVH 25165085 Ki = 1282 nM T08391 C8J4KL 25165278 Ki = 16 nM T08391 CRJ6M7 25165279 Ki > 1450 nM T08391 C7RBX0 25165280 Ki > 1450 nM T08391 CPEY29 25165481 Ki > 1450 nM T08391 C70DRX 25165482 Ki > 1450 nM T08391 CE8D1W 25165860 Ki = 1453 nM T08391 C6VZU2 25165861 Ki = 284 nM T08391 CT94MS 25166059 Ki > 1453 nM T08391 C5BM7F 25166250 Ki = 1450 nM T08391 C2D3FP 25167078 Ki > 1450 nM T08391 C8GL6I 25169133 IC50 < 3 nM T08391 C1G5JU 25169403 IC50 = 346 nM T08391 CZ28ES 25171661 IC50 < 3 nM T08391 CBIA60 25171662 IC50 = 4 nM T08391 C6ZTG4 25171663 IC50 < 3 nM T08391 CQH5N9 25171664 IC50 = 3 nM T08391 CQ04LW 25171665 IC50 < 3 nM T08391 CU9KV5 25171666 IC50 = 3 nM T08391 C0SE7H 25171874 IC50 < 3 nM T08391 C1YH8L 25171876 IC50 < 3 nM T08391 CC60NT 25171877 IC50 = 10 nM T08391 C8O1ZJ 25172085 IC50 < 3 nM T08391 CG6J5X 25172086 IC50 < 3 nM T08391 C0PX8V 25172087 IC50 = 33 nM T08391 C6UQG4 25181422 IC50 = 39 nM T08391 CX7CP9 25195487 IC50 = 200 nM T08391 CNG96H 25210579 IC50 > 10000 nM T08391 C0ZXH7 25236808 Ki = 2000 nM T08391 CC71QJ 27666048 IC50 > 100000 nM T08391 CT7X8Y 27700054 Ki > 3500 nM T08391 CW3QI4 42600633 Ki = 82.6 nM T08391 C92QDU 42611189 Ki = 86 nM T08391 CY4LG8 42622934 IC50 = 0.8 nM T08391 CAO2T4 42634832 Ki = 270 nM T08391 C57VJY 42635854 IC50 = 0.4 nM T08391 CP8RA7 42635855 IC50 = 1 nM T08391 C05BWT 42635901 IC50 = 1 nM T08391 CO9Y8F 42635906 IC50 = 11 nM T08391 CN1TI5 42635944 IC50 = 1 nM T08391 C5I9XW 42635949 IC50 = 2 nM T08391 CT63QC 42635982 IC50 = 95 nM T08391 CY5E4B 42635983 IC50 = 2 nM T08391 C8V6IK 42635984 IC50 = 3 nM T08391 C63HQD 42636016 IC50 = 2 nM T08391 C34DCR 42636018 IC50 = 2 nM T08391 CTOQ08 42636019 IC50 = 2 nM T08391 CU8MO6 42641406 IC50 = 6 nM T08391 CCB1E9 44124695 IC50 > 100000 nM T08391 CQI60M 44158549 IC50 = 6900 nM T08391 CBAN65 44158553 IC50 = 52 nM T08391 CH6OL2 44158658 IC50 = 3.4 nM T08391 CHD5N8 44158660 IC50 = 7.8 nM T08391 CU07NR 44158886 IC50 = 11 nM T08391 CLK7R8 44159000 IC50 = 0.5 nM T08391 CD0YP3 44159001 IC50 = 0.6 nM T08391 CQ8FJ4 44159590 IC50 = 3000 nM T08391 CY67LR 44159594 IC50 = 1.4 nM T08391 CZF1B5 44159711 IC50 = 1500 nM T08391 CQW4F1 44159839 IC50 = 34 nM T08391 CBK83A 44159959 IC50 = 22 nM T08391 CEF0X4 44159962 IC50 = 36 nM T08391 CBZ09W 44160079 IC50 = 560 nM T08391 C1ZY4N 44160207 IC50 = 0.2 nM T08391 CB0O2A 44186880 Ki = 1453 nM T08391 C9K7OP 44186882 Ki = 756 nM T08391 CX0ZU8 44186885 Ki = 1453 nM T08391 CNGV37 44189584 Ki > 1450 nM T08391 CIT2A7 44192904 IC50 = 76.7 nM T08391 C8KNA3 44219632 Ki > 4000 nM T08391 C0VIX4 44219633 Ki = 2400 nM T08391 CZB49P 44419474 IC50 = 19 nM T08391 CI9GX4 44419475 IC50 = 17 nM T08391 CAT2U0 44419478 IC50 = 68 nM T08391 CC36WM 44419481 IC50 = 113 nM T08391 C6BWA2 44419485 IC50 = 59 nM T08391 CXW0D5 44419491 IC50 = 4 nM T08391 CZY28V 44419492 IC50 = 8 nM T08391 CCM3W5 44419493 IC50 = 16 nM T08391 CG2R1T 44419498 IC50 = 51 nM T08391 C40WFE 44419499 IC50 = 153 nM T08391 CNZJ15 44419502 IC50 = 20 nM T08391 C5DL8E 44419515 IC50 > 10000 nM T08391 CMVY72 44419516 IC50 = 167 nM T08391 CNT03L 44419522 IC50 = 7218 nM T08391 CH46CM 44419523 IC50 = 51 nM T08391 CO20LA 44419524 IC50 = 12 nM T08391 C3CBQ4 44419526 IC50 = 49 nM T08391 C4XIY6 44419527 IC50 > 10000 nM T08391 CGH30Q 44419528 IC50 = 77 nM T08391 C42FJP 44419532 IC50 > 10000 nM T08391 C0FKV6 44419533 IC50 = 18 nM T08391 CXG7H4 44419544 IC50 = 56 nM T08391 CI2BL7 44419547 IC50 = 141 nM T08391 C2T5AQ 44419548 IC50 = 29 nM T08391 CT19AN 44419556 IC50 = 28 nM T08391 CE6T5F 44419559 IC50 = 7 nM T08391 CQ0Y6P 44432177 IC50 = 11 nM T08391 CSRD60 44432179 IC50 = 6 nM T08391 C1DZ5C 44432180 IC50 = 19 nM T08391 CWBI39 44432182 IC50 = 55 nM T08391 C73SGA 44432183 IC50 = 42 nM T08391 CA92GM 44432184 IC50 = 21 nM T08391 CTDI23 44432185 IC50 = 53 nM T08391 CI9NY3 44432187 IC50 = 25 nM T08391 CGFT15 44432188 IC50 = 222 nM T08391 CT0D6O 44432189 IC50 = 132 nM T08391 CFK94T 44432190 IC50 = 359 nM T08391 C3TG1J 44432191 IC50 = 323 nM T08391 CBO5P0 44432192 IC50 = 298 nM T08391 C2S8ZC 44432193 IC50 = 1860 nM T08391 CYH6P3 44520205 IC50 > 10000 nM T08391 CW2P1N 44555004 Ki = 1.7 nM T08391 C96QIW 44555963 Ki = 2 nM T08391 CP5M6H 44556110 Ki = 1.1 nM T08391 CQ18YJ 44556112 Ki = 0.6 nM T08391 C3VRO9 44557921 IC50 > 10000 nM T08391 COR3N9 44560358 IC50 = 572 nM T08391 CA69DI 44570386 IC50 = 9300 nM T08391 C8A2ZJ 44570387 IC50 = 1950 nM T08391 C0S8WJ 44570388 IC50 = 28600 nM T08391 CR7T0U 44570389 IC50 = 320 nM T08391 C5YL2S 44570390 IC50 = 370 nM T08391 CVC6A3 44570391 IC50 = 740 nM T08391 C5A8CV 44570392 IC50 = 5800 nM T08391 C6B3XH 44570434 IC50 = 8580 nM T08391 CS6MF4 44570435 IC50 = 3550 nM T08391 C45TSL 44570436 IC50 = 1950 nM T08391 CCRL12 44570437 IC50 = 3900 nM T08391 C0EC7O 44570438 IC50 = 1570 nM T08391 CF1Y6E 44570474 IC50 = 1110 nM T08391 C1JSB3 44570475 IC50 = 330 nM T08391 CRGC97 44570476 IC50 = 1220 nM T08391 C9B8UC 44570477 IC50 = 770 nM T08391 C8KQ9B 44605608 Ki = 210 nM T08391 C63WNF 44610370 IC50 = 1010 nM T08391 CT7V9E 44610371 IC50 = 319 nM T08391 CL40ZN 44610523 IC50 = 175 nM T08391 C6QT0J 44622837 IC50 > 1000 nM T08391 C9AVD2 44624425 Ki = 1.6 nM T08391 CKUA84 44626045 IC50 > 30000 nM T08391 C2SLI6 44631938 IC50 = 18 nM T08391 C4K8BX 45267171 IC50 = 33500 nM T08391 C25VIM 45267176 IC50 = 16900 nM T08391 C36DGY 45272290 IC50 > 40000 nM T08391 COT0W8 45272300 IC50 = 5100 nM T08391 CC79UA 45273165 IC50 > 40000 nM T08391 CNR8G6 45273175 IC50 > 40000 nM T08391 C4J5XF 45275254 IC50 = 4 nM T08391 CZ7T8F 45275363 IC50 = 15 nM T08391 CB58EO 45275368 IC50 = 27 nM T08391 CU3AD0 45275473 IC50 = 12 nM T08391 C7KMO9 45275580 IC50 = 3 nM T08391 CFN17Z 45280146 IC50 = 1.1 nM T08391 CA23WL 45280210 IC50 = 6 nM T08391 C96HCQ 45375954 IC50 = 56 nM T08391 CQ3KO2 45375955 IC50 = 1.2 nM T08391 C5G2MN 45375956 IC50 = 5 nM T08391 C6OX0V 45375974 IC50 < 3 nM T08391 C0QP2U 45483928 Ki = 260 nM T08391 CS7RO0 45483929 Ki = 480 nM T08391 CXF92W 45486106 IC50 = 200 nM T08391 CZXL23 45486109 IC50 = 44 nM T08391 CF8JM7 45486113 IC50 = 6500 nM T08391 CIE6V0 45486118 IC50 = 84 nM T08391 CV59GT 45486119 IC50 = 260 nM T08391 C9E0MS 45486120 IC50 = 4.7 nM T08391 C07DPA 45486121 IC50 = 4 nM T08391 CR7T9D 45486124 IC50 = 210 nM T08391 C7QK0X 45486129 IC50 = 880 nM T08391 CY36ZX 45486130 IC50 = 70 nM T08391 C04ZHY 45486136 IC50 = 50 nM T08391 C5SA2N 45486137 IC50 = 190 nM T08391 C91VMT 45486138 IC50 = 25 nM T08391 CLN7F0 45486139 IC50 = 3.1 nM T08391 C8RNJ5 45486142 IC50 = 270 nM T08391 C9FQJ4 45486147 IC50 = 87 nM T08391 CPM6O9 45486148 IC50 = 130 nM T08391 CX0HO6 45486156 IC50 < 3 nM T08391 CYZ13M 45486157 IC50 = 907 nM T08391 CZMD28 45486158 IC50 = 160 nM T08391 CMXY69 45486159 IC50 = 4.6 nM T08391 CA0O3Q 45486163 IC50 = 20 nM T08391 C5U1LS 45486164 Ki = 7 nM T08391 CN6G7A 45486168 IC50 = 4 nM T08391 CT9OP5 45486169 IC50 = 4666 nM T08391 C7D4GB 45486170 IC50 = 21 nM T08391 CET79H 45493316 IC50 = 110 nM T08391 CND6H4 46176417 IC50 = 120 nM T08391 CE45XW 46208354 IC50 = 4.9 nM T08391 CUHB49 46208355 IC50 = 4.1 nM T08391 CW38GO 46208357 IC50 = 5.5 nM T08391 C43COY 46208358 IC50 = 3.2 nM T08391 CE4Q7D 46208596 IC50 = 5.3 nM T08391 CM9UN7 46208601 IC50 = 1.1 nM T08391 CH7JB4 46209051 IC50 = 3.5 nM T08391 CY3HW5 46224684 IC50 > 10000 nM T08391 CLOZ21 46224796 Ki = 0.5 nM T08391 C9O2RG 46224797 Ki = 0.6 nM T08391 C9BET8 46224835 Ki = 13 nM T08391 C6TU1W 46224836 Ki = 42 nM T08391 C03MZI 46224837 Ki = 3 nM T08391 C9RGH2 46224876 Ki = 2100 nM T08391 C0C9IJ 46224910 Ki > 5000 nM T08391 CLPV83 46224911 Ki > 5000 nM T08391 CM8Z4P 46224912 Ki = 3800 nM T08391 CA4V3E 46224936 Ki = 1 nM T08391 CJ0P5D 46224938 Ki = 400 nM T08391 CVZ80Y 46224939 Ki = 4500 nM T08391 CG3SZ2 46224940 Ki > 5000 nM T08391 C3DJ5Q 46224970 Ki > 5000 nM T08391 C0NFE6 46224971 Ki = 29 nM T08391 C3R0EQ 46224972 Ki = 630 nM T08391 CI83TA 46224997 Ki = 34 nM T08391 C4VU8O 46224998 Ki = 3800 nM T08391 C86GDI 46225269 Ki = 2100 nM T08391 C9AJP4 46225270 Ki = 460 nM T08391 CV37ID 46225315 Ki = 1800 nM T08391 C1Z0JB 46225316 Ki = 370 nM T08391 CG6Y3N 46234403 IC50 = 234 nM T08391 C3JW8A 46234405 IC50 = 226 nM T08391 CWN3M0 46234565 EC50 = 2045 nM T08391 CLTU68 46234566 IC50 = 78 nM T08391 C5YH1F 46235625 IC50 = 47 nM T08391 CWLU63 46235938 IC50 = 181 nM T08391 CC25DT 46235942 IC50 = 7 nM T08391 CZ7J6K 46236109 IC50 = 48 nM T08391 C26NQY 46236112 IC50 = 92 nM T08391 C1S4LH 46398810 IC50 = 7.3 nM T08391 CG71EF 46832441 IC50 = 2 nM T08391 C1LNX9 46832443 IC50 = 5.5 nM T08391 CCK54P 46852509 IC50 = 85 nM T08391 CC57FP 46852510 IC50 = 8.9 nM T08391 C31UXV 46852812 IC50 = 13 nM T08391 COTJ39 46863083 IC50 = 13000 nM T08391 C35AIH 46865430 IC50 = 5 nM T08391 C2EK4B 46865431 IC50 = 5 nM T08391 CMZ0R3 46865529 IC50 = 4.3 nM T08391 C3B2NL 46865530 IC50 = 6.8 nM T08391 CC2O9R 46865656 IC50 = 1584.89 nM T08391 CJ3NV8 46865657 IC50 = 8 nM T08391 CQB16A 46872415 Ki = 3200 nM T08391 CLS29B 46872626 IC50 > 10000 nM T08391 C0AU7R 46879420 IC50 = 28 nM T08391 CUVG95 46879421 IC50 = 1550 nM T08391 CRZM17 46879422 IC50 = 170 nM T08391 CER6X5 46879423 IC50 = 97 nM T08391 C7O1AZ 46879483 IC50 = 500 nM T08391 C2DU1O 46879484 IC50 = 95 nM T08391 CB31AL 46879485 IC50 = 285 nM T08391 C5URZ1 46879545 IC50 = 840 nM T08391 C3LEW4 46879546 IC50 = 7000 nM T08391 CKI4M6 46880119 IC50 = 3250 nM T08391 CU8KB7 46880120 IC50 = 1800 nM T08391 C47OXF 46880121 IC50 = 560 nM T08391 CK87XC 46880122 IC50 = 3400 nM T08391 CC3Y7B 46880193 IC50 = 393 nM T08391 C0GS1C 46880194 IC50 = 470 nM T08391 CV9IL3 46880195 IC50 = 1000 nM T08391 C0M5ND 46880196 IC50 = 270 nM T08391 C60UAN 46880197 IC50 = 320 nM T08391 C5NZ8R 46880686 IC50 = 150 nM T08391 CZ79VE 46880687 IC50 = 8 nM T08391 C0YNH6 46880737 IC50 < 3 nM T08391 CGO7C5 46880738 IC50 = 14 nM T08391 C75ZTG 46880739 IC50 = 39 nM T08391 C9T7WL 46880784 IC50 = 8 nM T08391 CSV4G2 46880785 IC50 = 5 nM T08391 CS6W4P 46882359 IC50 = 467 nM T08391 CF5B9A 46882360 IC50 = 322 nM T08391 CX4UK2 46882361 IC50 = 202 nM T08391 C5FNK6 46882409 IC50 = 83 nM T08391 CN8OR4 46882410 IC50 = 81 nM T08391 CEI25D 46882411 IC50 = 33 nM T08391 CJZ8H9 46882412 IC50 = 16 nM T08391 C6Z4KW 46882470 IC50 = 6 nM T08391 CH0Y5K 46882471 IC50 = 11 nM T08391 C70LVA 46882472 IC50 = 8 nM T08391 CP1BH3 46882539 IC50 = 12 nM T08391 CQR25C 46882540 IC50 = 9 nM T08391 CVTO81 46882541 IC50 = 16 nM T08391 CQ6T0Y 46882542 IC50 = 14 nM T08391 COV4E6 46882589 IC50 = 18 nM T08391 CDG2N8 46882590 IC50 = 2 nM T08391 C0UX2M 46882591 IC50 = 4 nM T08391 CN0I6Z 46882592 IC50 = 6 nM T08391 CZ7A9N 46882802 IC50 = 69 nM T08391 CCK7H2 46882803 IC50 = 47 nM T08391 C9MW2L 46885052 IC50 = 4200 nM T08391 C69HUW 46885053 IC50 = 101 nM T08391 CASL67 46885231 IC50 = 685 nM T08391 CEU6O4 46885232 IC50 = 501 nM T08391 CE27LI 46885233 IC50 = 7.1 nM T08391 CB8LN4 46885234 IC50 = 13 nM T08391 CMX7U6 46885289 IC50 = 12.5 nM T08391 CB1ZN5 46885290 IC50 = 3.1 nM T08391 C2O8RZ 46886323 IC50 > 1000 nM T08391 C60GAV 46929544 IC50 > 8000 nM T08391 CP34VL 46929748 IC50 > 1000 nM T08391 CJ2E9Q 46929857 IC50 > 25000 nM T08391 CCN08S 46934144 IC50 = 106700 nM T08391 CT7EY8 49817363 IC50 = 330 nM T08391 CBP75U 49838138 IC50 = 0.9 nM T08391 CMKB24 49838268 IC50 = 3 nM T08391 CF0UM2 49838516 IC50 = 0.64 nM T08391 CTJX98 49838518 IC50 = 1.4 nM T08391 CSE4K3 49838775 IC50 = 1.27 nM T08391 CB34CO 49839441 Ki = 35 nM T08391 C2DGY0 49839445 Ki > 3500 nM T08391 C06MKW 49839561 Ki = 27.6 nM T08391 CT3SH4 49839838 IC50 = 3 nM T08391 CF91RS 49843531 IC50 > 10000 nM T08391 C7A6IZ 49850211 EC50 > 20000 nM T08391 C57FQH 49856318 IC50 = 790 nM T08391 C70QSD 49856319 IC50 = 510 nM T08391 C24SMN 49856320 IC50 = 1440 nM T08391 CHK7D3 49856321 IC50 = 480 nM T08391 CK4LJ5 49856703 Ki = 770 nM T08391 CZVU24 49856845 Ki = 0.3 nM T08391 C9J7LZ 49857227 Ki = 7.1 nM T08391 CS72TM 49859752 IC50 = 1.8 nM T08391 CK5TH3 50906783 EC50 = 2800 nM T08391 CA0WR3 50914031 IC50 = 250 nM T08391 CQE9D1 50925411 IC50 = 578 nM T08391 C64HTN 50925513 IC50 = 1 nM T08391 C2Y6QS 50938552 IC50 > 10000 nM T08391 CF26MU 50991562 IC50 = 33 nM T08391 CHS63D 50993724 IC50 < 3 nM T08391 C2SKV4 50993725 IC50 = 9 nM T08391 CKN2H7 50993726 IC50 = 16 nM T08391 CMH3A2 50993881 IC50 < 3 nM T08391 C20VEP 50994284 IC50 > 10000 nM T08391 CI1L0M 50994285 IC50 = 4700 nM T08391 C7ZWT8 50994286 IC50 = 9150 nM T08391 C6VNE1 50994366 IC50 = 1444 nM T08391 CSEZ73 50994367 IC50 > 10000 nM T08391 C1R8ZI 50995341 IC50 = 129 nM T08391 C53NRD 50995522 IC50 = 180 nM T08391 CAZQ43 51003133 IC50 > 1000 nM T08391 CWKS75 51003514 IC50 = 1 nM T08391 C9NYP4 51036677 IC50 > 10000 nM T08391 C4WRY3 51037112 IC50 > 10000 nM T08391 CRI28Z 51037948 IC50 > 10000 nM T08391 CDU4Q5 51346827 Ki = 898 nM T08391 CXA03W 52920796 IC50 > 100 nM T08391 CEQN27 52936621 Ki = 370 nM T08391 C1PLW9 52941200 IC50 = 1400 nM T08391 CA9DE6 52941228 IC50 > 10000 nM T08391 CR2QD0 52941284 IC50 = 8350 nM T08391 C1T5EH 52942437 IC50 > 10000 nM T08391 C54UKL 52942449 IC50 = 3940 nM T08391 CO8W1R 52942701 IC50 = 55 nM T08391 CY20GZ 52942702 IC50 = 274 nM T08391 CEPS91 52943663 IC50 = 5000 nM T08391 C2IQ5B 52943672 IC50 > 10000 nM T08391 CMP9W8 52944434 IC50 = 139 nM T08391 CTN0C3 52944839 IC50 > 10000 nM T08391 CXG0B3 52946111 IC50 = 3157 nM T08391 CN2Q0G 52946313 IC50 = 14 nM T08391 CT2U3E 52947304 IC50 = 2500 nM T08391 CU49PE 52947324 IC50 = 11500 nM T08391 C1QWK5 52947390 IC50 = 512 nM T08391 CY42JP 52947547 IC50 = 200 nM T08391 C7S8TB 52948490 IC50 = 29000 nM T08391 CQY9D0 52948526 IC50 = 2110 nM T08391 C8TC3P 52948550 IC50 = 2500 nM T08391 CIM43G 52948562 IC50 > 10000 nM T08391 CWG31A 52948678 IC50 = 4 nM T08391 CQ87RP 52949754 IC50 = 11800 nM T08391 CNW53F 52949761 IC50 = 630 nM T08391 C6VHI5 52949798 IC50 = 26 nM T08391 C2XNP3 53024548 IC50 = 12200 nM T08391 CR36JQ 53232414 IC50 = 115300 nM T08391 C93WOC 53232452 IC50 < 3 nM T08391 C6OTY5 53251320 IC50 = 11000 nM T08391 CZ71UE 53316996 IC50 = 190 nM T08391 CE5Y7P 53316997 IC50 = 110 nM T08391 CH13DY 53316998 IC50 = 22 nM T08391 CXO42U 53317010 IC50 = 5.3 nM T08391 C3HT4Y 53317607 IC50 = 2 nM T08391 CH3Y2L 53317729 IC50 = 14000 nM T08391 C8KXF6 53317730 IC50 = 22 nM T08391 CE8OY2 53317913 IC50 > 100 nM T08391 CI8PJ6 53318277 IC50 = 2700 nM T08391 C7T2RG 53318278 IC50 = 2.2 nM T08391 C4RBZ8 53318283 IC50 = 3.5 nM T08391 C7D4IR 53318284 IC50 = 4.6 nM T08391 CZS8K4 53319042 Ki = 791 nM T08391 CGRX02 53319638 IC50 = 31 nM T08391 C6QP8W 53319646 IC50 = 7.3 nM T08391 C8OAH1 53319647 IC50 = 0.6 nM T08391 C5ZT4W 53319648 IC50 = 2.4 nM T08391 CUD21V 53320263 Ki = 644 nM T08391 C76DUB 53320946 IC50 = 4.8 nM T08391 C0XZA6 53320947 IC50 = 1.2 nM T08391 CF4LM9 53321614 IC50 = 2.8 nM T08391 CFHD02 53322268 IC50 = 59 nM T08391 CESA85 53323614 Ki = 281 nM T08391 C39GZV 53323629 IC50 = 1.1 nM T08391 C2W9OA 53324451 IC50 > 10000 nM T08391 C8M9WN 53324904 IC50 = 4.5 nM T08391 CU6W1L 53324912 IC50 = 2.1 nM T08391 CB94UN 53326192 IC50 = 9.3 nM T08391 CVY30S 53326193 IC50 = 3 nM T08391 CEF6L2 53326206 IC50 = 0.9 nM T08391 CQS1R8 53341008 Ki = 28 nM T08391 CNPM14 53341082 IC50 > 3000 nM T08391 C4BM5W 53341107 Ki = 12 nM T08391 CZKQ72 53341161 Ki = 53 nM T08391 CN59SH 53341248 Ki = 10 nM T08391 CB83XH 53341368 Ki = 56 nM T08391 CD2CH6 53341413 Ki = 40 nM T08391 CGP23R 53341457 Ki = 1.2 nM T08391 C0SWH5 53348216 IC50 > 40000 nM T08391 C8ZRE3 53356518 IC50 = 3068 nM T08391 C95JTI 53373594 Ki = 6.5 nM T08391 C8NA4L 53384644 IC50 > 30000 nM T08391 C56TYK 53385837 IC50 = 121.6 nM T08391 CNLM53 53385838 IC50 = 123.1 nM T08391 C1XE2K 53385938 IC50 = 345.4 nM T08391 C37JTE 53385939 IC50 = 37 nM T08391 CV92IB 53386254 IC50 = 18 nM T08391 CU6QF7 53386309 IC50 < 0.6 nM T08391 CYU0R4 53386418 IC50 = 0.5 nM T08391 C7RM6Q 53386421 IC50 < 0.3 nM T08391 CEN91X 53389820 IC50 = 231.2 nM T08391 C24FQU 53465297 IC50 = 379 nM T08391 CM12OQ 53475998 Ki = 130 nM T08391 C6W0PN 53476000 Ki = 2100 nM T08391 C4G2ST 53476104 Ki = 95 nM T08391 C37PHN 53497571 IC50 = 3940 nM T08391 CCF1B3 53497572 IC50 = 1 nM T08391 COF6B0 54577892 IC50 = 0.17 nM T08391 C2ECL9 54577896 IC50 = 1.6 nM T08391 CY5C8A 54589404 IC50 = 0.8 nM T08391 CS7E0A 54672927 IC50 = 106.2 nM T08391 CHZ27O 54673255 IC50 = 22.4 nM T08391 C7X5ZM 54673258 IC50 = 44.3 nM T08391 CZ84NW 54673259 IC50 = 10.8 nM T08391 CX0U2A 54673422 IC50 = 32.6 nM T08391 C19FZK 54673425 IC50 = 355.2 nM T08391 CBPT15 54673763 IC50 = 1010 nM T08391 C36BAI 54673911 IC50 = 10.9 nM T08391 CD8ZK6 54674056 IC50 = 70 nM T08391 CFTE97 54674369 IC50 = 250 nM T08391 CUCI05 54674990 IC50 = 43 nM T08391 CH0IM9 54754557 IC50 = 0.7 nM T08391 C1ZF5H 54754832 Ki > 3200 nM T08391 CY9KA8 54755181 Ki > 3200 nM T08391 CE1ZK6 54759168 IC50 > 10000 nM T08391 C1XS2J 54760383 IC50 = 1200 nM T08391 CXH2P4 54766274 IC50 = 74 nM T08391 CD28VZ 54766423 IC50 = 100 nM T08391 CAP1J7 54766425 IC50 = 340 nM T08391 C75JFM 54766426 IC50 = 800 nM T08391 CDIC43 54766427 IC50 = 77 nM T08391 C2XDG1 54766428 IC50 = 380 nM T08391 C0XCY1 54766576 IC50 = 75 nM T08391 CPH3Y7 54766578 IC50 = 190 nM T08391 C0T4SL 54766726 IC50 = 83 nM T08391 CZD70Q 54767039 IC50 = 4.8 nM T08391 CN1DZ6 54767189 IC50 = 5.4 nM T08391 C83VCG 56587966 IC50 = 91 nM T08391 C1W3EZ 56591424 IC50 = 0.6 nM T08391 CTB63S 56591428 IC50 = 13 nM T08391 CWR1P6 56591446 IC50 = 0.8 nM T08391 C6ZL7H 56592816 IC50 = 81 nM T08391 C6Z1QA 56592817 IC50 = 1.2 nM T08391 C9IY4P 56594654 IC50 = 100 nM T08391 CG4E7C 56594655 IC50 = 19 nM T08391 C21GRJ 56594656 IC50 = 2700 nM T08391 CD7FW6 56594657 IC50 = 59 nM T08391 C67KYZ 56594658 IC50 = 23 nM T08391 CN96IU 56594659 IC50 = 110 nM T08391 CWYN98 56594660 IC50 = 70 nM T08391 CVDL32 56594786 IC50 = 180 nM T08391 CSE7W1 56594788 IC50 = 13 nM T08391 C0FCD9 56594790 IC50 = 23 nM T08391 CKZ27O 56594916 IC50 = 9 nM T08391 CR70XD 56595052 IC50 = 3 nM T08391 C3DJO1 56595053 IC50 = 12 nM T08391 C8KO5T 56595054 IC50 = 4 nM T08391 CW4QC9 56595056 IC50 = 8 nM T08391 C5KR6N 56595558 Ki = 67 nM T08391 COI9U2 56595687 Ki > 4000 nM T08391 C2AM6B 56595688 Ki > 4000 nM T08391 CFY2I4 56595689 Ki > 4000 nM T08391 CAM8E1 56595690 Ki = 590 nM T08391 CN5EV7 56595691 Ki > 4000 nM T08391 C6ET0W 56595693 Ki > 4000 nM T08391 CM8JX1 56604907 IC50 = 1000 nM T08391 CTR10F 56658543 Ki > 4000 nM T08391 C9HQ6G 56659204 IC50 = 12 nM T08391 C1FA3D 56659205 IC50 = 1100 nM T08391 C2E7VD 56666167 IC50 = 12 nM T08391 CGF4J3 56666168 IC50 = 14 nM T08391 CEH31Y 56668417 IC50 = 0.2 nM T08391 CG3Z0E 56669566 IC50 = 10 nM T08391 CC73NZ 56676392 IC50 = 5 nM T08391 CR23VJ 56679727 IC50 = 13 nM T08391 CXF9T4 56679728 IC50 = 41 nM T08391 CY1QA2 56683053 IC50 = 370 nM T08391 CR9A5O 56834874 IC50 = 2400 nM T08391 C58MSV 56834889 IC50 = 1620 nM T08391 CUT2G8 56835062 IC50 = 2.5 nM T08391 CJBL48 56925034 IC50 = 50 nM T08391 CBFR12 56925356 IC50 = 48 nM T08391 C80DRA 56925357 IC50 = 72 nM T08391 C0HUN8 56925358 IC50 = 100 nM T08391 C6Z2EA 56925359 IC50 = 1170 nM T08391 CC1MN2 56925454 IC50 = 1170 nM T08391 C3XC0T 56925455 IC50 = 27 nM T08391 CBW6T3 56925456 IC50 = 10 nM T08391 C8G3NO 56925457 IC50 = 2890 nM T08391 CHS19C 56925458 IC50 = 1370 nM T08391 CBMO42 56925459 IC50 = 8 nM T08391 CQTD41 56925550 IC50 = 135 nM T08391 CI9T3S 56925551 IC50 = 5 nM T08391 CS84ZU 56925552 IC50 = 4720 nM T08391 C9IVD0 56929216 Ki = 12 nM T08391 C0BO4X 56934550 Ki = 62 nM T08391 C5FY9U 56945728 IC50 = 250 nM T08391 C7D0EY 56946378 IC50 = 1700 nM T08391 CUQ50W 56946379 IC50 = 18 nM T08391 C3B2YH 56951311 IC50 = 0.17 nM T08391 CJMB49 56953110 Ki = 26 nM T08391 CAK91L 56955954 IC50 > 3600 nM T08391 CSO40C 56973425 Ki = 4.4 nM T08391 CU5BD9 57336812 IC50 = 1.8 nM T08391 C31LJU 57339437 Ki = 200 nM T08391 CMF7J0 57339438 Ki = 250 nM T08391 CPO2J4 57342178 IC50 = 150 nM T08391 C72PED 57342179 IC50 = 63 nM T08391 CA93PN 57342180 IC50 = 370 nM T08391 CI70CT 57345538 IC50 = 650 nM T08391 CVS76D 57390492 IC50 = 0.5 nM T08391 C4P5YQ 57390669 IC50 = 0.54 nM T08391 C3N2SF 57390670 IC50 = 1.1 nM T08391 COV39R 57390671 IC50 = 0.5 nM T08391 C9MW1O 57390672 IC50 = 0.3 nM T08391 CBJ93Q 57390673 IC50 = 0.4 nM T08391 C10WYL 57390861 IC50 = 16 nM T08391 CC7LW5 57392473 IC50 = 0.23 nM T08391 CEDR08 57392474 IC50 = 1 nM T08391 C79QPH 57392475 IC50 = 0.5 nM T08391 CS2R7J 57392476 IC50 = 0.36 nM T08391 C5O1HP 57392676 IC50 = 2.1 nM T08391 C6SKR3 57392677 IC50 = 6.3 nM T08391 C16RBI 57393424 IC50 = 450 nM T08391 C56DZN 57394024 IC50 = 0.6 nM T08391 C93GNJ 57394178 IC50 = 0.33 nM T08391 CZI79U 57394179 IC50 = 1.2 nM T08391 C0ZSA5 57394180 IC50 = 0.4 nM T08391 C3J4NV 57394381 IC50 = 2 nM T08391 CK74ND 57394382 IC50 = 0.22 nM T08391 C43EQN 57394383 IC50 = 0.52 nM T08391 C1V9MC 57394384 IC50 = 16 nM T08391 CKS67A 57396146 IC50 = 0.22 nM T08391 CE4FA1 57396924 IC50 = 330 nM T08391 CWJ70D 57397964 IC50 = 62 nM T08391 CAQ9D6 57397965 IC50 = 2900 nM T08391 CE8JW3 57398441 IC50 = 1.5 nM T08391 CFU5H3 57399413 IC50 = 2.1 nM T08391 C8CTY7 57399414 IC50 = 0.47 nM T08391 CKE7L0 57399415 IC50 = 0.35 nM T08391 C8BD2Q 57399416 IC50 = 480 nM T08391 CZX8R7 57399606 IC50 = 0.09 nM T08391 CMU89A 57401172 IC50 = 3.7 nM T08391 C43NFS 57401173 IC50 = 1 nM T08391 CL9Z2D 57401363 IC50 = 0.64 nM T08391 C8F4ME 57401364 IC50 = 0.27 nM T08391 CZTG84 57402768 IC50 = 0.9 nM T08391 CK06MA 57402935 IC50 = 1.14 nM T08391 CZ85FM 57402936 IC50 = 0.5 nM T08391 C9WMS3 57402937 IC50 = 0.8 nM T08391 C0FS4C 57402938 IC50 = 0.35 nM T08391 C9GN1M 57403118 IC50 = 0.6 nM T08391 C56CSP 57403119 IC50 = 39 nM T08391 C6A8WC 57502370 IC50 = 2132 nM T08391 CIO15D 57502371 IC50 > 10000 nM T08391 C6YOU9 57502372 IC50 = 1406 nM T08391 C8DN1A 57502373 IC50 = 2874 nM T08391 C15XOS 57502374 IC50 = 2165 nM T08391 CEF53Z 57502376 IC50 = 47 nM T08391 CTY54N 57502377 IC50 = 136 nM T08391 CBLN61 57502378 IC50 = 8 nM T08391 CDV4R1 57502379 IC50 = 1.5 nM T08391 CILJ54 57502380 IC50 = 1615 nM T08391 CS90RX 57502381 IC50 = 3 nM T08391 CE6B7C 57502382 IC50 = 0.8 nM T08391 CC82QJ 57502383 IC50 = 3.1 nM T08391 C72OWZ 57502386 IC50 = 1.1 nM T08391 CHC90Q 57502387 IC50 = 1.4 nM T08391 C9Z6QJ 57502388 IC50 = 0.7 nM T08391 CMF31G 57502390 IC50 = 26 nM T08391 C4QXU9 57514090 IC50 = 193 nM T08391 C0YW2D 57514091 IC50 = 5.6 nM T08391 CU8Y3P 57514092 IC50 = 1.3 nM T08391 C5K3VZ 57514093 IC50 = 4 nM T08391 CNQ6K8 57659282 IC50 = 617 nM T08391 CS75LF 57659335 IC50 = 20 nM T08391 COU4M1 57915982 IC50 = 17 nM T08391 C1G5SK 57916044 IC50 = 23 nM T08391 C3C0PQ 57916049 IC50 = 43 nM T08391 CH6RB0 57916164 IC50 = 23 nM T08391 C9MF8U 57928260 IC50 = 11 nM T08391 C3KQJ8 57928435 IC50 = 1.7 nM T08391 C5H8VE 57928583 IC50 = 11 nM T08391 C13VIO 57928632 IC50 = 120 nM T08391 C8BTO7 57928826 IC50 = 5 nM T08391 C18MVX 57990771 IC50 = 5000 nM T08391 C4TQ9L 57990797 IC50 = 5.7 nM T08391 C4XC3V 57990957 IC50 > 980 nM T08391 CB6F5S 57990969 IC50 = 0.9 nM T08391 C13BGJ 57991037 IC50 = 7.9 nM T08391 CDRB84 57991074 IC50 = 129.9 nM T08391 CJ4B2L 57991089 IC50 = 621.7 nM T08391 C9EA1S 57991186 IC50 = 1431.3 nM T08391 C5B3HI 57991212 IC50 = 2.9 nM T08391 C48LZT 57991260 IC50 > 980 nM T08391 C8R4FE 57991377 IC50 = 2.2 nM T08391 C19UKS 57991389 IC50 = 5.2 nM T08391 C1KH5D 57991398 IC50 = 1.7 nM T08391 CSN47V 57991473 IC50 = 8.7 nM T08391 CD6ZP3 58009815 EC50 = 1600 nM T08391 CWU1Y3 58009825 EC50 = 890 nM T08391 C8S6MY 58010054 EC50 = 4200 nM T08391 CM1B4V 58010265 EC50 = 4800 nM T08391 CGR87Y 58063067 Ki = 1.3 nM T08391 C3J7XM 58063084 Ki = 1 nM T08391 CW2Z5I 58063100 Ki = 0.3 nM T08391 C1EVX0 58063117 Ki = 0.1 nM T08391 C7NE0H 58063121 Ki = 0.1 nM T08391 COT5L0 58063146 Ki = 1.6 nM T08391 CGBY54 58063225 Ki = 1 nM T08391 C1RF4W 58063241 Ki = 31.9 nM T08391 C0P8VW 58063334 Ki = 2.5 nM T08391 CZO2J1 58063487 Ki = 5.1 nM T08391 C2U5TY 58063491 Ki = 1.8 nM T08391 CQND09 58177229 IC50 = 102 nM T08391 CU4I8X 58177247 IC50 = 71 nM T08391 CLEH36 58177279 IC50 = 54 nM T08391 CIK3U8 58177332 IC50 = 36 nM T08391 C8D2TA 58177362 IC50 = 181 nM T08391 CYC85B 58177456 IC50 = 9 nM T08391 C7BU0H 58180518 IC50 = 3.1 nM T08391 CKA28H 58180521 IC50 = 1.2 nM T08391 C2I5LO 58180525 IC50 = 2.1 nM T08391 CN4OZ8 58180573 IC50 = 1.4 nM T08391 C92FOB 58180591 IC50 = 0.9 nM T08391 CWXC70 58180596 IC50 = 2.5 nM T08391 C9N1QB 58180623 IC50 = 1.5 nM T08391 CSK1U8 58180628 IC50 = 1.4 nM T08391 C6LT9S 58180630 IC50 = 1.9 nM T08391 CCBT87 58180639 IC50 = 1.4 nM T08391 C7Q8YZ 58374808 IC50 > 10000 nM T08391 CP81TW 58394456 Ki = 59 nM T08391 C4H3FY 58394522 Ki = 20 nM T08391 CM6SK2 58394565 Ki = 32 nM T08391 C6HPO3 58394632 Ki = 15 nM T08391 CK71MA 58394722 Ki = 580 nM T08391 CO5TH6 58394820 Ki = 47 nM T08391 CY0UV6 58394828 Ki = 2.9 nM T08391 CW7D0O 58394866 Ki = 21 nM T08391 C0W2AT 58394878 Ki = 669 nM T08391 C97QAK 58394904 Ki = 18 nM T08391 C9Q4WD 58394916 Ki = 25 nM T08391 CI37CQ 58394927 Ki = 5 nM T08391 C5RGU7 58394946 Ki = 721 nM T08391 C6KO0G 58395044 IC50 = 5700 nM T08391 CDK5L1 58395223 Ki = 3.8 nM T08391 C9J5UV 58395232 Ki = 11 nM T08391 CYC87B 58395253 Ki = 487 nM T08391 C5S8BK 58395290 Ki = 66 nM T08391 C4H2ZP 58395301 Ki = 8.3 nM T08391 C28ADB 58395446 Ki = 2.1 nM T08391 CLA5V3 58395468 Ki = 121 nM T08391 C0X5CV 58395476 Ki = 3.7 nM T08391 C9TV2G 58398904 IC50 = 490 nM T08391 CR9T7W 58438557 IC50 = 2030 nM T08391 CY3W6B 58438580 IC50 = 134.2 nM T08391 CR7C4V 58438607 IC50 = 0.8 nM T08391 C9MIL7 58450666 IC50 = 203 nM T08391 CWX4G9 58522116 IC50 = 2320 nM T08391 C4A6LT 58522124 IC50 = 1710 nM T08391 CI9VB0 58522237 IC50 = 580 nM T08391 C1LE9A 58522238 IC50 = 900 nM T08391 C74ACR 58522276 IC50 = 1000 nM T08391 CI0L1J 58522322 IC50 = 1210 nM T08391 CVMO97 58522377 IC50 = 1250 nM T08391 C7S1PR 58522381 IC50 = 410 nM T08391 C2W0OD 58539094 Ki > 3200 nM T08391 C6CDB7 58539140 Ki = 3000 nM T08391 CB3TQ8 58539146 Ki > 3200 nM T08391 C7WRQ5 58539268 Ki > 3200 nM T08391 C97ZGJ 58539301 Ki > 3200 nM T08391 C8X6YE 58557497 IC50 = 11400 nM T08391 CX0Q2W 58688109 IC50 = 804 nM T08391 C6BPR2 58985201 IC50 > 30000 nM T08391 C3YHW8 59186181 Ki = 5 nM T08391 C5MHP0 59186191 Ki = 4.8 nM T08391 CSR49F 59186194 Ki = 17.7 nM T08391 CT8CI4 59186216 Ki = 19.3 nM T08391 CGS2D4 59186263 Ki = 3 nM T08391 CHG45P 59186268 Ki = 0.6 nM T08391 C8NA2Z 59186270 Ki = 40.6 nM T08391 C2AF7G 59186271 Ki = 70.9 nM T08391 CI93GZ 59186442 Ki = 9.1 nM T08391 C4XQ9E 59186482 Ki = 2 nM T08391 CS07KJ 59186487 Ki = 0.9 nM T08391 CD30LA 59186489 Ki = 0.3 nM T08391 CGRE28 59198979 Ki = 0.5 nM T08391 CG4Y8K 59198994 Ki = 0.5 nM T08391 C4TJS9 59199010 Ki = 0.4 nM T08391 CPD28H 59199061 Ki = 1.4 nM T08391 CJA50L 59199121 Ki = 0.7 nM T08391 C3S1CI 59199131 Ki = 0.6 nM T08391 CR6UM8 59199136 Ki = 1.1 nM T08391 CR2OB1 59199142 Ki = 0.6 nM T08391 C6TAW4 59199165 Ki = 0.5 nM T08391 CPWM60 59291925 IC50 = 12 nM T08391 C3CV0R 59291929 IC50 = 46 nM T08391 COXI75 59291940 IC50 = 370 nM T08391 CE6KO4 59291951 IC50 = 17 nM T08391 CT3EW2 59292007 IC50 = 3.2 nM T08391 C2PE0T 59292008 IC50 = 41 nM T08391 CU3W2S 59292043 IC50 = 49 nM T08391 CC6J4I 59363349 EC50 = 452 nM T08391 CQ93TM 59363383 EC50 = 778 nM T08391 CKQ31B 59363409 EC50 = 798 nM T08391 CZ3TG1 59375154 IC50 = 212 nM T08391 CU7Q5A 59435986 IC50 = 2 nM T08391 C64IHJ 59435987 IC50 = 7 nM T08391 C2VG8U 59436001 IC50 = 1 nM T08391 CCJ81A 59436022 IC50 = 37 nM T08391 CG9NO0 59436049 IC50 = 0.9 nM T08391 CT4P2H 59436062 IC50 = 0.8 nM T08391 C7T9PR 59436066 IC50 = 0.15 nM T08391 C8D5BA 59436080 IC50 = 9 nM T08391 CRV24D 59436099 IC50 = 3 nM T08391 CP9BH2 59436109 IC50 = 0.5 nM T08391 C81AOP 59525628 IC50 = 178 nM T08391 CI0G2S 59525684 IC50 = 93 nM T08391 C3R7ZX 59525688 IC50 = 140 nM T08391 CP3SN6 59525717 IC50 = 36 nM T08391 CT35BZ 59525728 IC50 = 690 nM T08391 CVD4E5 59525760 IC50 = 80 nM T08391 CP1F6X 59526007 IC50 = 380 nM T08391 CM7OV6 59526068 IC50 = 155 nM T08391 C4N9MS 59526260 IC50 = 312 nM T08391 CFEU09 59589639 Ki = 207 nM T08391 C0DV7R 59589757 Ki = 59 nM T08391 CMPO72 59599420 IC50 = 215 nM T08391 CXJ63M 59603829 IC50 = 1200 nM T08391 CQEU96 59603842 IC50 = 64 nM T08391 CDMO01 59617921 Ki > 3500 nM T08391 CUNY05 59617942 Ki > 3500 nM T08391 CY7V3I 59617971 Ki = 1400 nM T08391 CM6B3E 59618010 Ki = 380 nM T08391 CQCG48 59618036 Ki = 2500 nM T08391 CJ5GF1 59618081 Ki > 3500 nM T08391 CT12JO 59618117 Ki = 860 nM T08391 C42OZL 59618123 Ki = 55 nM T08391 COI26N 59618146 Ki > 3500 nM T08391 CR5GJ4 59618147 Ki = 1300 nM T08391 C9GB1C 59618160 Ki = 2400 nM T08391 CR9F7D 59618164 Ki = 310 nM T08391 C7XWE2 59618171 Ki = 510 nM T08391 C2EIA3 59618285 Ki = 130 nM T08391 C1ZKR9 59618313 Ki = 2900 nM T08391 C26BNV 59618424 Ki = 2700 nM T08391 C3B7CU 59618428 Ki = 63 nM T08391 CBH83T 59618445 Ki = 60 nM T08391 C3HC4P 59618462 Ki = 2400 nM T08391 CX0FQ2 59618505 Ki = 20 nM T08391 CG8ET4 59618513 Ki = 250 nM T08391 CR27IT 59618564 Ki > 3500 nM T08391 CSZA16 60155724 IC50 > 3600 nM T08391 CNY59P 60165955 Ki = 0.3 nM T08391 CY3QT8 60165956 Ki = 25 nM T08391 CKT4Y7 60170769 Ki = 6.4 nM T08391 C3YSV5 60170770 Ki = 74 nM T08391 C34RVN 60170771 Ki = 9.3 nM T08391 C74FPI 60170772 Ki = 11 nM T08391 CTC8E4 60170773 Ki = 17 nM T08391 CR80CH 60170858 Ki = 12 nM T08391 C3PA9G 60170859 Ki = 21 nM T08391 C2AEG3 60170860 Ki = 520 nM T08391 CHJM71 60170861 Ki = 26 nM T08391 CBP48G 60170862 Ki = 28 nM T08391 C3R0NO 63107904 IC50 = 3960 nM T08391 CK6WO0 66552478 IC50 < 10000 nM T08391 CE4RV7 66558256 IC50 > 10000 nM T08391 CQK4Y2 66570958 IC50 = 8 nM T08391 C5RAC8 66571005 IC50 = 12 nM T08391 CVXT19 66571006 IC50 = 308 nM T08391 C5UFY3 66571008 IC50 = 3 nM T08391 CG8AP3 66571009 IC50 = 187 nM T08391 C20EXP 66571075 IC50 = 24 nM T08391 C3WF4H 66571076 IC50 = 10 nM T08391 C3IRH5 66571077 IC50 = 150 nM T08391 CYS96O 66571078 IC50 = 21 nM T08391 CPW01U 66571135 IC50 = 2 nM T08391 C32BMH 66571136 IC50 = 53 nM T08391 CC04XH 66571138 IC50 = 35 nM T08391 CI6A2Z 66571139 IC50 = 109 nM T08391 CGP12A 66571140 IC50 = 57 nM T08391 CJL68E 66571195 IC50 = 46 nM T08391 C6STC7 66571196 IC50 = 247 nM T08391 C3U6ED 66571199 IC50 = 268 nM T08391 CQ49JM 66571200 IC50 = 114 nM T08391 CY3P8G 66571201 IC50 = 3056 nM T08391 CYFL93 66571254 IC50 = 44 nM T08391 C5H1VS 66571255 IC50 = 154 nM T08391 CG3XE8 66571256 IC50 = 384 nM T08391 C3WM6R 66571316 IC50 = 43 nM T08391 C8DSK2 66571317 IC50 = 1235 nM T08391 C72WVF 66571377 IC50 = 66 nM T08391 C9T4VJ 66571378 IC50 = 1537 nM T08391 CJ08ZL 66604045 IC50 = 5.7 nM T08391 CY0I2V 66604274 IC50 = 370 nM T08391 CD0LJ6 66604359 IC50 = 2.4 nM T08391 CS8HK2 66604394 IC50 = 120 nM T08391 C7U8GC 66604464 IC50 = 110 nM T08391 CXU94O 66604576 IC50 = 17 nM T08391 CE9T0V 66604664 IC50 = 86 nM T08391 C7WO4A 66604791 IC50 = 3.1 nM T08391 CW53KR 66604810 IC50 = 130 nM T08391 CNW05G 66604855 IC50 = 6.8 nM T08391 CT4RU2 66604890 IC50 = 1.7 nM T08391 C0JS8O 66604914 IC50 = 1.2 nM T08391 CW9LD1 66604921 IC50 = 8 nM T08391 CTMX20 66605009 IC50 = 7.4 nM T08391 C0EVU7 66605043 IC50 = 27 nM T08391 CP0DB1 66605115 IC50 = 10.2 nM T08391 CGS8J2 66605151 IC50 = 4.3 nM T08391 CB1WC9 66605298 IC50 = 3.5 nM T08391 CCWU74 66605322 IC50 = 16 nM T08391 C7Q8ZG 66605359 IC50 = 7.4 nM T08391 C16TEK 66605475 IC50 = 6.1 nM T08391 C7MOJ6 66605487 IC50 = 470 nM T08391 CDZA70 66605639 IC50 = 5.2 nM T08391 C53NBQ 66605756 IC50 = 280 nM T08391 CN5BR8 66605844 IC50 = 2.6 nM T08391 CDES25 66606401 IC50 = 6.2 nM T08391 C5J4MR 66850717 Ki = 3.2 nM T08391 CC6JF4 66851197 Ki = 3.2 nM T08391 CO2H4Q 66851201 Ki = 49 nM T08391 C3BTX2 66851307 Ki = 41.2 nM T08391 C7ONK1 66851426 Ki = 2.1 nM T08391 C5PVB2 67008690 IC50 = 194 nM T08391 C8OZ6W 67008828 IC50 = 84 nM T08391 C1HSE0 67035086 IC50 = 1100 nM T08391 CWI6K5 67035106 IC50 > 10000 nM T08391 C38RGB 67035556 IC50 > 10000 nM T08391 CZX1E0 67123420 IC50 = 68 nM T08391 C0RCI2 67123577 IC50 = 0.3 nM T08391 C37NKO 67129970 IC50 = 4920 nM T08391 CK80LJ 67130050 IC50 = 4170 nM T08391 CV63UL 67240318 IC50 > 10000 nM T08391 C6YHJ5 67277266 IC50 = 430 nM T08391 C78TXA 67277273 IC50 = 200 nM T08391 C0O7TC 67277276 IC50 = 2.6 nM T08391 C3YK7Q 67277763 IC50 = 310 nM T08391 CQXW93 67277840 IC50 = 850 nM T08391 CF4AB0 67277979 IC50 = 1800 nM T08391 CFM39N 67278030 IC50 = 640 nM T08391 C5U2IW 67278045 IC50 = 23 nM T08391 CS9K0L 67278047 IC50 = 140 nM T08391 C2FW8H 67278142 IC50 = 85 nM T08391 CQRS42 67278151 IC50 = 82 nM T08391 C5V9DZ 67278165 IC50 = 500 nM T08391 CMJ29W 67278195 IC50 = 88 nM T08391 C2C7BD 67278380 IC50 = 190 nM T08391 CVL35U 67278385 IC50 = 97 nM T08391 CKVB79 67278425 IC50 = 17 nM T08391 C2C1RE 67329237 IC50 > 30000 nM T08391 CV80IQ 67330694 IC50 = 27 nM T08391 C16THB 67351896 Ki = 27 nM T08391 CFX84K 67352945 Ki = 21 nM T08391 C1FLT6 67354280 Ki = 401 nM T08391 CEF67O 67383086 Ki = 14 nM T08391 CLO13H 67383145 Ki = 110 nM T08391 C94UAF 67383148 Ki = 43 nM T08391 C5D2QA 67383227 Ki = 93 nM T08391 C4AE8Z 67383253 Ki = 10 nM T08391 CW8Q3F 67383552 Ki = 5.4 nM T08391 C6UF3T 67383612 Ki = 21 nM T08391 CV38SD 67383669 Ki = 440 nM T08391 C9WY2P 67383875 Ki = 22 nM T08391 CJ2Q1S 67383893 Ki = 26 nM T08391 CUK87J 67387753 Ki = 150 nM T08391 C14RKJ 67479440 IC50 > 100000 nM T08391 C5WQC2 67502257 IC50 > 1000 nM T08391 CZ0O6N 68234726 Ki = 16 nM T08391 CA89HR 68235185 Ki = 490 nM T08391 CYR38C 68241014 IC50 = 400 nM T08391 C0MY1I 68241371 IC50 = 130 nM T08391 CX6S4E 68254533 IC50 = 800 nM T08391 C4U1IR 68291322 IC50 = 42 nM T08391 C2P7DB 68291391 IC50 = 280 nM T08391 CRM3S0 68291627 IC50 = 210 nM T08391 C4LKB3 68291752 IC50 = 18 nM T08391 CQ49HB 68291755 IC50 = 70 nM T08391 CXI4L1 68291797 IC50 = 170 nM T08391 C8T5VB 68291830 IC50 = 62 nM T08391 CPRW18 68291866 IC50 = 438 nM T08391 C6UWI3 68291981 IC50 = 130 nM T08391 CYN89R 68292156 IC50 = 120 nM T08391 C76EZC 68292170 IC50 = 130 nM T08391 CGA0W6 68292183 IC50 = 31 nM T08391 C93LZT 68292196 IC50 = 130 nM T08391 C8I7GC 68293638 IC50 > 10000 nM T08391 CD56XK 68293660 IC50 > 10000 nM T08391 CYI75G 68678653 IC50 > 30000 nM T08391 C7GRV2 68755406 IC50 = 2320 nM T08391 CIL58T 69023801 IC50 = 12.8 nM T08391 C5DGR9 69036886 IC50 = 1173 nM T08391 CK8DC3 69046862 IC50 = 15 nM T08391 CV0K3P 69267827 IC50 = 4 nM T08391 CVH5M3 69671224 Ki = 190 nM T08391 COX56A 69809432 IC50 = 45 nM T08391 CECG39 69809726 IC50 = 108 nM T08391 C7FA5L 69811602 EC50 = 3690 nM T08391 C92EAC 69811936 EC50 = 2665 nM T08391 C0XO1M 69812740 IC50 = 82 nM T08391 CJ96RN 70099013 Ki > 3200 nM T08391 CRZ5V2 70495652 Ki = 63.3 nM T08391 CS47OP 70496411 Ki = 11.9 nM T08391 CV0NP6 70496595 Ki = 0.4 nM T08391 CK5H1Y 70497007 Ki = 103 nM T08391 CTG78Y 70497097 Ki = 5.6 nM T08391 CTY17Z 70497535 Ki = 16.7 nM T08391 C6NSG3 70497750 Ki = 9.7 nM T08391 CWP52K 70497865 Ki = 15.5 nM T08391 CP48DJ 70498203 Ki = 41.1 nM T08391 CQH47T 70498861 Ki = 14 nM T08391 C7VJ6A 70647728 IC50 = 370 nM T08391 CASQ98 70650259 IC50 = 90 nM T08391 CQ2F8J 70824464 Ki = 610 nM T08391 CBF3Q6 71042865 IC50 = 972 nM T08391 CNR2Y9 71061323 IC50 = 1.3 nM T08391 C51JTW 71061588 IC50 = 1.7 nM T08391 CF69WT 71061828 IC50 = 3.6 nM T08391 COU2C5 71061858 IC50 = 7.4 nM T08391 CW9OE6 71061878 IC50 = 2 nM T08391 CK9LZ3 71061981 IC50 = 1.9 nM T08391 CU1T4P 71061987 IC50 = 5.3 nM T08391 CJH94D 71062030 IC50 = 1.5 nM T08391 CUW46K 71062043 IC50 = 4.3 nM T08391 C05VNE 71062076 IC50 = 4.8 nM T08391 C4AC9U 71212257 IC50 < 0.2 nM T08391 COD6B2 71222450 Ki = 34 nM T08391 COR71Z 71285696 IC50 = 740 nM T08391 C3ZL5S 71285760 IC50 = 56 nM T08391 CME92O 71285933 IC50 = 15 nM T08391 C2FL6H 71286084 IC50 = 1.3 nM T08391 C14YOJ 71286184 IC50 = 13 nM T08391 CX23BP 71288497 IC50 = 20 nM T08391 CH1AJ3 71288512 IC50 = 1.1 nM T08391 CA1T5H 71288539 IC50 = 16 nM T08391 CYU2Z4 71288594 IC50 = 28 nM T08391 CBY4K0 71288602 IC50 = 22 nM T08391 CWLC45 71288607 IC50 = 38 nM T08391 CDST08 71288618 IC50 = 10800 nM T08391 C45HTF 71288693 IC50 = 3.3 nM T08391 COC20B 71288707 IC50 = 83 nM T08391 C6JD3S 71288724 IC50 = 4.2 nM T08391 COV78A 71288729 IC50 = 5.9 nM T08391 C8DY1N 71288732 IC50 = 57 nM T08391 CNV7B6 71300296 Ki = 0.72 nM T08391 C49STX 71450071 Ki = 5.2 nM T08391 CX4LE5 71453548 Ki = 7 nM T08391 CPO7Y1 71454973 Ki = 12 nM T08391 CAN57Z 71455263 Ki > 3200 nM T08391 CKT60L 71455860 Ki = 920 nM T08391 C4D1TQ 71456076 IC50 > 980 nM T08391 CPY5K3 71457046 Ki > 3200 nM T08391 C1X6YV 71457047 Ki = 3 nM T08391 CML7F1 71458913 Ki = 64 nM T08391 CFN35P 71459077 Ki = 0.6 nM T08391 CR6O7Q 71462440 Ki > 3200 nM T08391 C01XHF 71510730 IC50 = 392 nM T08391 C09YSR 71510731 IC50 = 594 nM T08391 C9DIK2 71512060 IC50 > 10000 nM T08391 CCN01X 71547862 IC50 > 10000 nM T08391 CVEO06 71558636 IC50 = 39 nM T08391 C07SFW 71600166 IC50 = 1350 nM T08391 CWJ1G4 71600167 IC50 = 446 nM T08391 CKY79O 71615499 Ki = 1.41 nM T08391 C8GLY0 71615500 IC50 = 4 nM T08391 CA7Q3S 71615501 IC50 = 3 nM T08391 CVYS15 71617859 IC50 = 3.2 nM T08391 C7T5LI 71655637 Ki = 1232 nM T08391 CT3M4B 71655638 Ki = 446 nM T08391 CSC81X 71655639 Ki = 57 nM T08391 C3U1ZV 71655709 Ki = 17 nM T08391 CE1JQ3 71655774 Ki = 33 nM T08391 CX5OU4 71681533 Ki = 18 nM T08391 C29FVT 71681534 Ki = 90 nM T08391 C7WQP2 71681535 Ki = 76 nM T08391 CEQM71 71681536 EC50 > 10 nM T08391 CV5FB0 71681691 Ki = 44 nM T08391 C6JH7K 71681692 Ki = 49 nM T08391 CS62NH 71698376 IC50 = 111900 nM T08391 CI8X1R 71698379 IC50 = 138200 nM T08391 C5QK6S 71727668 IC50 = 26 nM T08391 C8PSM2 71737832 Ki = 145 nM T08391 CO76WG 71818715 Ki = 8 nM T08391 CR02FG 71818862 Ki = 2200 nM T08391 CY6WE7 71818863 Ki = 2200 nM T08391 CW52BU 71943288 IC50 = 2380 nM T08391 C54XWG 72190869 IC50 > 10000 nM T08391 C4XY6C 72195599 IC50 = 126 nM T08391 CLD12K 72201823 IC50 = 2.7 nM T08391 CYQN46 72201826 IC50 = 4.1 nM T08391 CP9CJ3 72201957 IC50 = 164 nM T08391 CMVI93 72201958 IC50 = 37.9 nM T08391 CD9Z4H 72202092 IC50 = 3.7 nM T08391 CLIS85 72202093 IC50 = 9.4 nM T08391 C5Q7YT 72202095 IC50 = 12.1 nM T08391 C8NGE4 72202097 IC50 = 42.9 nM T08391 C1W6LK 72202246 IC50 = 55.4 nM T08391 C6W4ZS 72202247 IC50 = 4.2 nM T08391 C1N7LQ 72202249 IC50 = 0.5 nM T08391 C2W6TI 72202397 IC50 = 1.6 nM T08391 CIKL36 72202398 IC50 = 9.6 nM T08391 C1I4LX 72202399 IC50 = 3125 nM T08391 C4CB2S 72202400 IC50 = 53.7 nM T08391 CVI63X 72202547 IC50 = 1.6 nM T08391 C0EZ3I 72202548 IC50 = 2.9 nM T08391 C7OY3V 72202549 IC50 = 14.2 nM T08391 CH40KC 72202550 IC50 = 9.2 nM T08391 CA5CI3 72202825 IC50 = 6.4 nM T08391 C6THF4 72374600 Ki = 70 nM T08391 CHK46S 72375658 Ki = 123 nM T08391 COPS30 72375659 Ki = 377 nM T08391 CB9ZL4 72375660 Ki = 130 nM T08391 C0K5IO 72375661 Ki = 54 nM T08391 C7PG8Z 72375662 Ki = 189 nM T08391 CCZO42 72375759 Ki = 550 nM T08391 CEV9X5 72375760 Ki = 201 nM T08391 COE6R4 72375761 Ki = 766 nM T08391 C1G8RD 72375763 Ki = 690 nM T08391 C8SLE9 72375764 Ki = 380 nM T08391 C74WLS 72375765 Ki = 3200 nM T08391 CP2KL5 72375766 Ki = 3200 nM T08391 CT9D3J 72375844 Ki = 1500 nM T08391 CZN81X 72375845 Ki = 567 nM T08391 CXL52K 72375846 Ki = 1400 nM T08391 CAV52F 72375847 Ki = 575 nM T08391 C3QT2E 72375850 Ki = 63 nM T08391 C0UJ9M 72375852 Ki = 150 nM T08391 CNJ03L 72375990 Ki > 3500 nM T08391 C5R0WV 72375991 Ki = 3200 nM T08391 CVUL48 72375992 Ki = 1800 nM T08391 CO8KW2 72375993 Ki > 3500 nM T08391 CN0I2W 72375994 Ki > 3500 nM T08391 C1XD7U 72375995 Ki = 3100 nM T08391 C8BJ4U 72375996 Ki > 3500 nM T08391 C7XFW2 72375997 Ki > 3500 nM T08391 CJB95D 72375998 Ki > 3500 nM T08391 CS5V9L 72376089 Ki = 1400 nM T08391 C37GPL 72376090 Ki = 2000 nM T08391 C9U3WO 72376091 Ki > 3500 nM T08391 C0DL3F 72698602 IC50 < 1 nM T08391 CK7F6U 72700776 Ki = 1 nM T08391 CLOE10 72706962 IC50 = 575 nM T08391 C1D2AM 72737634 IC50 = 1 nM T08391 CG16YE 72771106 IC50 = 460 nM T08391 CMK8Z4 73055651 IC50 = 3 nM T08391 C50CRU 73056517 IC50 = 1 nM T08391 CQAI18 73056519 IC50 = 12 nM T08391 C16AQK 73056520 IC50 = 8 nM T08391 C2ZFQ1 73057136 IC50 = 16 nM T08391 CH43OS 73057443 IC50 = 1 nM T08391 CDS4T9 73057444 IC50 = 20 nM T08391 CXD38C 73346480 Ki = 0.6 nM T08391 C0G5RD 73347974 Ki = 574 nM T08391 CRAW59 73349195 Ki = 230 nM T08391 C41ZJV 73349520 Ki = 1.8 nM T08391 CJE73Y 73352545 Ki = 23 nM T08391 CPRD59 73352546 Ki = 9 nM T08391 C4BUW7 73353407 IC50 = 20 nM T08391 CXT70E 73354035 Ki = 13 nM T08391 CGI13D 73354036 Ki = 158 nM T08391 CL4SD8 73355260 Ki > 3500 nM T08391 CMR72H 73355566 Ki = 21 nM T08391 CPT46O 73355567 Ki > 5600 nM T08391 C04CXF 73355568 Ki = 59 nM T08391 C3G2BM 73357112 Ki = 3 nM T08391 CO6F2B 73357113 Ki = 4 nM T08391 C8DSE2 75108379 IC50 < 3 nM T08391 CS41CX 75108409 IC50 = 33 nM T08391 CH20VA 75108447 IC50 = 24 nM T08391 CP90QE 75108517 IC50 < 3 nM T08391 CG6T5S 76072368 IC50 = 425.6 nM T08391 COMF95 76072369 IC50 = 10.8 nM T08391 CRK1L2 76210601 IC50 = 22 nM T08391 CO0BQ5 76310565 IC50 = 1480 nM T08391 C6ZAB2 76310566 IC50 > 10000 nM T08391 C0F6VU 76310567 IC50 > 10000 nM T08391 CDO38G 76310568 IC50 > 10000 nM T08391 CL42BQ 76310569 IC50 > 10000 nM T08391 CWI1Q4 76310570 IC50 = 1238 nM T08391 C8OY6Q 76310785 IC50 > 100000 nM T08391 CAL3U7 76310788 IC50 > 100000 nM T08391 C7SXJ1 76314208 IC50 = 1270 nM T08391 CSDI71 76314209 IC50 = 490 nM T08391 C12YAE 76314414 IC50 > 100000 nM T08391 CM6LI3 76314606 IC50 = 0.6 nM T08391 CXF1I3 76317774 IC50 > 10000 nM T08391 CY79VS 76317775 IC50 > 10000 nM T08391 CNK2I1 76317776 IC50 > 10000 nM T08391 CS02NA 76317777 IC50 = 1637 nM T08391 CAHW32 76317778 IC50 = 1270 nM T08391 CT9JM4 76317888 IC50 = 670 nM T08391 C97RBS 76317979 IC50 > 100000 nM T08391 C2SMK1 76321491 IC50 > 10000 nM T08391 C2DSX7 76321492 IC50 = 10080 nM T08391 CI2VZ6 76321886 IC50 = 26 nM T08391 CL0T7B 76322219 IC50 = 21513 nM T08391 CXA4O1 76325093 IC50 > 10000 nM T08391 CEZ64F 76325209 IC50 = 50 nM T08391 C1AI0J 76325315 IC50 > 100000 nM T08391 CPQA45 76325323 IC50 > 100000 nM T08391 C8GK0H 76328659 IC50 > 10000 nM T08391 C74RUX 76329058 IC50 = 10 nM T08391 CJN89E 76332335 IC50 > 10000 nM T08391 CW1QK4 76332336 IC50 = 2130 nM T08391 C2P1MX 76332338 IC50 = 11080 nM T08391 CB5Y0Z 76332540 IC50 > 100000 nM T08391 CB4KQ7 76335967 IC50 > 10000 nM T08391 C84PFQ 76335968 IC50 = 9687 nM T08391 CW1HQ9 76370451 IC50 = 5 nM T08391 CD6Y1F 78320046 IC50 = 550 nM T08391 CW08SU 78320048 IC50 = 220 nM T08391 CWI93D 78323836 IC50 = 381 nM T08391 C5UK9L 78323837 IC50 = 542 nM T08391 CQ3EJ1 78324132 IC50 = 6810 nM T08391 C7VOX0 78324136 IC50 = 1196 nM T08391 CA2Y8L 78324435 IC50 = 1090 nM T08391 C4I7WD 78324744 IC50 = 412 nM T08391 CQ2SU8 78673832 IC50 > 30000 nM T08391 CE0W9R 78673833 IC50 > 30000 nM T08391 CNI6U3 86267948 IC50 = 442 nM T08391 CV8UZ1 86278565 IC50 = 225 nM T08391 CZ97VP 86294733 IC50 = 680 nM T08391 CPG3A5 86302574 IC50 = 21052 nM T08391 C96EDF 86660048 IC50 = 7100 nM T08391 CC8I0M 86707711 IC50 = 15 nM T08391 CW4Z2F 89470642 IC50 = 1.2 nM T08391 CBRF87 89470690 IC50 = 2.8 nM T08391 C7B8OH 89470730 IC50 = 0.47 nM T08391 CDQ8C6 89471114 IC50 = 1.5 nM T08391 C4G5LP 89471136 IC50 = 3 nM T08391 CU6J4F 89498235 Ki = 23 nM T08391 CS7GX8 89708625 IC50 = 162400 nM T08391 C1HW4B 89735655 IC50 = 4400 nM T08391 CG9C6J 89765129 IC50 = 0.7 nM T08391 C13GOX 89775209 IC50 = 180 nM T08391 C3N6RU 89775221 IC50 = 70 nM T08391 C69JXR 90034304 IC50 = 131 nM T08391 CDO6N1 90034309 IC50 = 85 nM T08391 C3VJ2W 90034362 IC50 = 620 nM T08391 CB74RS 90034368 IC50 = 71 nM T08391 CE8T5K 90034382 IC50 = 690 nM T08391 CFX7M4 90034390 IC50 = 73 nM T08391 CEG3A4 90035164 IC50 = 9 nM T08391 CG5P9A 90153688 IC50 > 50000 nM T08391 CV64KY 90183363 IC50 > 1000 nM T08391 CL4JO2 90183809 IC50 = 718 nM T08391 CTV52A 90367281 IC50 = 19 nM T08391 CFB75T 90479825 IC50 = 6 nM T08391 CY0UC4 90645194 IC50 > 10000 nM T08391 CV9H8U 90656285 IC50 = 1500 nM T08391 CG7E1U 90656286 IC50 = 1225 nM T08391 CDF9O2 90656287 IC50 = 300 nM T08391 C7EXH8 91755097 IC50 = 11 nM T08391 C37IZB 91755098 IC50 = 140 nM T08391 C7UAK5 91809175 IC50 > 2000 nM T08391 C8RG6H 91827514 IC50 = 40 nM T08391 CVR1I7 91827515 IC50 = 8.2 nM T08391 CAU45T 91971978 IC50 > 30000 nM T08391 C64SIO 92042864 IC50 = 1050 nM T08391 C9BL4M 92045136 IC50 > 22000 nM T08391 CXU1Z2 101043725 IC50 > 2000 nM T08391 CRI0S4 101891768 IC50 > 1000 nM T08391 C9G5TC 102515538 Ki = 9 nM T08391 CM2C3W 105539869 IC50 = 1700 nM T08391 CU4O5Z 112901888 IC50 = 140 nM T08391 C3ECY5 117625437 IC50 = 14 nM T08391 CZC84D 117769161 IC50 = 27 nM T08391 CE7BZ8 117769174 IC50 = 160 nM T08391 CBJ07Q 117769217 IC50 = 70 nM T08391 CXHQ08 117769229 IC50 = 15 nM T08391 CS9WO4 117769234 IC50 = 11 nM T08391 C61VXQ 117769241 IC50 = 15 nM T08391 C1SA9I 117769244 IC50 = 19 nM T08391 C0VY7C 117769271 IC50 = 20 nM T08391 C6O9BT 117769272 IC50 = 47 nM T08391 CSR9B0 117769289 IC50 = 20 nM T08391 C2M9CR 117769307 IC50 = 38 nM T08391 C7FWS3 117769309 IC50 = 7.3 nM T08391 CYWV32 117769339 IC50 = 29 nM T08391 CZV35K 117769346 IC50 = 21 nM T08391 C5V6RG 117769349 IC50 = 80 nM T08391 C4O1PX 117769362 IC50 = 22 nM T08391 CPV4C8 117769365 IC50 = 15 nM T08391 CP3MC5 117769379 IC50 = 17 nM T08391 C8V6LG 117769392 IC50 = 22 nM T08391 C2NBZ8 117769396 IC50 = 17 nM T08391 COV59Y 117769408 IC50 = 49 nM T08391 CXJ3I6 117769409 IC50 = 30 nM T08391 C8LTZ6 117769464 IC50 = 19 nM T08391 C4KL1Y 117769470 IC50 = 14 nM T08391 CQ46WT 117769476 IC50 = 36 nM T08391 CSKO30 117769533 IC50 = 44 nM T08391 C6XC3W 117769575 IC50 = 9 nM T08391 CS95HO 117769592 IC50 = 27 nM T08391 C0PIL5 117769623 IC50 = 25 nM T08391 CO3DA2 117769866 IC50 = 7 nM T08391 CI46CP 117770056 IC50 = 390 nM T08391 C7NI8L 117770083 IC50 = 140 nM T08391 CJ3QC8 117770200 IC50 > 10000 nM T08391 CSD47C 117770482 IC50 = 13 nM T08391 C8SNB9 117770595 IC50 = 910 nM T08391 CJ1V9A 117770654 IC50 = 550 nM T08391 CS8E6M 117770678 IC50 = 1400 nM T08391 CM7X9N 117770754 IC50 = 310 nM T08391 C4CFG6 117770831 IC50 = 830 nM T08391 C0X1EQ 117809257 IC50 = 31 nM T08391 CDUH09 117809287 IC50 = 3.5 nM T08391 C8HYU9 117926195 IC50 > 10000 nM T08391 CGQK96 118115537 IC50 > 10000 nM T08391 C2OX1Q 118115706 IC50 = 2030 nM T08391 CWCO47 118115913 IC50 > 10000 nM T08391 C72LYV 118116131 IC50 > 10000 nM T08391 C4JW5D 118116385 IC50 > 10000 nM T08391 CY0H6Z 118129292 IC50 = 68 nM T08391 CJ1LF6 118129295 IC50 = 331 nM T08391 CA7FL8 118129378 IC50 = 2910 nM T08391 C7ZM6W 118129401 IC50 = 369 nM T08391 CNX7M9 118473558 IC50 > 2000 nM T08391 CK6Z8O 118475621 IC50 = 107 nM T08391 CIVS69 118475644 IC50 = 32 nM T08391 C17FYA 118475649 IC50 = 351 nM T08391 CE49ZI 118475652 IC50 = 51 nM T08391 C65NIK 118475658 IC50 > 3000 nM T08391 C0A9RJ 118475705 IC50 = 17.6 nM T08391 CWQ36P 118475893 IC50 > 3000 nM T08391 CN04RH 118475894 IC50 = 945 nM T08391 C2P0CG 118475938 IC50 = 421 nM T08391 CJYV54 118494221 IC50 = 82.4 nM T08391 CLTV08 118690376 IC50 = 17 nM T08391 CRK6J2 118690573 IC50 = 13 nM T08391 CTR74C 118690690 IC50 = 12 nM T08391 CY7BI2 118706214 IC50 > 10000 nM T08391 C2C0AG 118707521 IC50 > 100000 nM T08391 C2DJA0 118707522 IC50 > 100000 nM T08391 CBF28W 118707523 IC50 > 100000 nM T08391 CQ6ON4 118707525 IC50 > 100000 nM T08391 C38UWP 118707526 IC50 > 100000 nM T08391 C64ZQX 118707543 IC50 > 100000 nM T08391 C7EG0V 118712812 IC50 = 394 nM T08391 C57YED 118712813 IC50 = 59 nM T08391 CX58DI 118716791 IC50 > 30000 nM T08391 CD9X2B 118716796 IC50 > 30000 nM T08391 C2YJ0O 118716797 IC50 > 30000 nM T08391 CL3UO9 118716798 IC50 > 30000 nM T08391 C71BAM 118716799 IC50 > 30000 nM T08391 CU4EL6 118716806 IC50 > 30000 nM T08391 CI5W9H 118720010 IC50 = 44 nM T08391 COQ9S4 118720011 IC50 > 1000 nM T08391 CP0IO9 118722564 IC50 = 4410 nM T08391 C5K2QD 118723914 IC50 = 30 nM T08391 C59YJC 118723915 IC50 = 16 nM T08391 C2ON7Y 118723916 IC50 = 570 nM T08391 C5U8WG 118723917 IC50 = 130 nM T08391 C0ZMR8 118723918 IC50 = 100 nM T08391 C4Z5LJ 118723919 IC50 = 350 nM T08391 C85ELI 118723920 IC50 = 61 nM T08391 CGW49X 118723921 IC50 = 150 nM T08391 CXC8K9 118723922 IC50 = 400 nM T08391 CR5JD8 118723923 IC50 = 110 nM T08391 C9W1BU 118723924 IC50 = 380 nM T08391 CW2G9E 118724201 IC50 > 30000 nM T08391 CXQM59 118727237 IC50 = 8500 nM T08391 C1XE3V 118727239 IC50 = 9500 nM T08391 CU0BP1 118727245 IC50 = 6900 nM T08391 CHT6K9 118728811 Ki > 4000 nM T08391 CUA3Y2 118728812 Ki > 4000 nM T08391 CDQ78G 118728813 Ki = 620 nM T08391 CZ6XL7 118728814 Ki = 270 nM T08391 CMO67K 118728815 Ki = 200 nM T08391 CR2M0Q 118728816 Ki > 4000 nM T08391 C62SCL 118728817 Ki > 4000 nM T08391 CSB30C 118728819 Ki = 840 nM T08391 CV7XU8 118728820 Ki = 390 nM T08391 C3J1EX 118728821 Ki > 4000 nM T08391 CIWB78 118728822 Ki = 1100 nM T08391 CP18SE 118728823 Ki = 240 nM T08391 CM42CA 118728824 Ki > 4000 nM T08391 C9Q7CL 118728825 Ki > 4000 nM T08391 CCR3S0 118728826 Ki = 740 nM T08391 C5NIL4 118729140 IC50 = 1068 nM T08391 C6TP4G 118729141 IC50 = 950 nM T08391 CQJY72 118729142 IC50 = 220 nM T08391 CWNA60 118729861 IC50 = 216 nM T08391 CN2SA5 118734641 IC50 = 293 nM T08391 CF6J5Q 118734642 IC50 = 1044 nM T08391 CMHF86 118734643 IC50 = 686 nM T08391 CUE83V 118734644 IC50 = 246 nM T08391 C67IDL 118734645 IC50 = 558 nM T08391 CFD82L 118734646 IC50 = 1475 nM T08391 C26ZJS 118734647 IC50 = 613 nM T08391 CM5A9U 118734648 IC50 = 547 nM T08391 C7HP6N 118734649 IC50 = 684 nM T08391 CVIN49 118734650 IC50 = 835 nM T08391 CQCX41 118737057 IC50 = 2911 nM T08391 C8JGN7 118868847 IC50 = 888 nM T08391 C3DK1Q 118868914 IC50 = 156 nM T08391 CQ1TL7 118879520 IC50 = 286 nM T08391 CAZO34 118911466 IC50 = 11000 nM T08391 C6VAE4 118911477 IC50 = 51 nM T08391 CRQV39 118911480 IC50 = 130 nM T08391 C5Z0XH 118911481 IC50 = 410 nM T08391 CG0T1W 118911482 IC50 = 2800 nM T08391 COD91F 118911483 IC50 = 15000 nM T08391 C5LYI2 118911484 IC50 = 7800 nM T08391 CA9P3K 118911491 IC50 = 260 nM T08391 CB81YO 118911492 IC50 = 66 nM T08391 C2DG5M 118911497 IC50 = 30000 nM T08391 CI2EU5 118911501 IC50 = 7400 nM T08391 CA3EF6 118911506 IC50 = 160 nM T08391 C9BE2G 118911507 IC50 = 16000 nM T08391 C75DOY 118911508 IC50 = 1400 nM T08391 CZ3D0U 118911512 IC50 = 11000 nM T08391 C1AE4J 118911514 IC50 = 1300 nM T08391 CN53SL 118911517 IC50 = 250 nM T08391 CCX4J8 118911542 IC50 = 1300 nM T08391 C7R0NJ 118911545 IC50 = 4700 nM T08391 CIS3Z5 118911549 IC50 = 5.5 nM T08391 C49PME 118911551 IC50 = 9100 nM T08391 CJT3P9 118911552 IC50 = 98000 nM T08391 CX01BU 118911553 IC50 = 1200 nM T08391 C0TU7V 118911556 IC50 = 470 nM T08391 C0TX7B 118911557 IC50 = 1000 nM T08391 CYI3O6 118911558 IC50 = 150 nM T08391 C28MLV 118911560 IC50 = 930 nM T08391 C49UGI 118911561 IC50 = 1200 nM T08391 C9LD1H 118911562 IC50 = 4500 nM T08391 CTR8D0 118911563 IC50 = 1100 nM T08391 CY5EN8 118911565 IC50 = 30 nM T08391 C84BPW 118911566 IC50 = 36 nM T08391 CT4MJ8 118911570 IC50 = 59 nM T08391 C2AZP5 118911571 IC50 = 1100 nM T08391 C2S7MO 118911575 IC50 = 50 nM T08391 C45HFX 118911579 IC50 = 9100 nM T08391 CCSH64 118911580 IC50 = 6300 nM T08391 CB48OQ 118911581 IC50 = 420 nM T08391 CZY2V6 118911582 IC50 = 13000 nM T08391 C2PA8M 118911583 IC50 = 97 nM T08391 C70XKA 118911584 IC50 = 2500 nM T08391 CD9C1A 118911585 IC50 = 2800 nM T08391 CRZ20W 118911587 IC50 = 180 nM T08391 CTQ4J9 118911588 IC50 = 180 nM T08391 C3QKH8 118911601 IC50 = 150 nM T08391 COY26N 118911635 IC50 = 6500 nM T08391 CL3C9A 118911638 IC50 = 4400 nM T08391 CN4O2C 118911639 IC50 = 480 nM T08391 C9O4WL 118911640 IC50 = 2800 nM T08391 C3SE0K 118911642 IC50 = 1300 nM T08391 C5LHC4 118911643 IC50 = 8.4 nM T08391 CYTV80 121284861 IC50 > 2000 nM T08391 C37DUM 121293882 IC50 > 2000 nM T08391 CXQR89 121294143 IC50 = 1100 nM T08391 C08KEM 122179540 IC50 = 4700 nM T08391 C3AJ4C 122179546 IC50 = 6700 nM T08391 CG0RP7 122179547 IC50 = 2700 nM T08391 C1A0SQ 122179548 IC50 = 5600 nM T08391 C42GSX 122180520 Ki > 4000 nM T08391 CO7D4I 122182021 IC50 = 1300 nM T08391 CY9M5S 122182022 IC50 = 7.3 nM T08391 C2MCH6 122182157 IC50 = 84 nM T08391 CD92SA 122182158 IC50 = 640 nM T08391 CK4A6L 122182159 IC50 = 14 nM T08391 C9OWX5 122186256 IC50 > 10000 nM T08391 C3J6BA 122186261 IC50 > 10000 nM T08391 CZN2V0 122188510 IC50 = 6864 nM T08391 CD62MC 122191616 IC50 = 4.5 nM T08391 CJI3E4 122191617 IC50 = 14 nM T08391 CFU15S 122191618 IC50 = 4.2 nM T08391 CE4F3A 122191619 IC50 = 25 nM T08391 CAC5U1 122191620 IC50 = 210 nM T08391 C8C1PI 122191621 IC50 = 1300 nM T08391 CA0D5W 122191622 IC50 = 570 nM T08391 CZ9K5C 122191623 IC50 = 43 nM T08391 C3NYR0 122191624 IC50 = 450 nM T08391 CRF2K0 122191625 IC50 = 230 nM T08391 CFKD32 122191637 IC50 = 1020 nM T08391 CPY1K9 122191778 IC50 = 2451 nM T08391 C1H4IX 122192065 IC50 = 2200 nM T08391 C98EJO 122192066 IC50 = 20500 nM T08391 CM1XD7 122192067 IC50 = 2900 nM T08391 C0MLH5 122192068 IC50 = 1600 nM T08391 CC4T6A 122192069 IC50 = 3200 nM T08391 CGO6M7 122192070 IC50 = 4100 nM T08391 CBP34K 122192071 IC50 = 2800 nM T08391 CA2TF6 122192072 IC50 = 2700 nM T08391 CFY30Z 122192073 IC50 = 2600 nM T08391 CJ09XF 122192074 IC50 = 2600 nM T08391 C6LS8X 122192075 IC50 = 5900 nM T08391 C7DJA5 122192076 IC50 = 4800 nM T08391 CAS86F 122192079 IC50 = 13500 nM T08391 CG7TP0 122192080 IC50 = 4700 nM T08391 C5K8UM 122192081 IC50 = 1600 nM T08391 CS4XB9 122199230 IC50 = 11900 nM T08391 CNA45R 122362931 IC50 = 113 nM T08391 CV7RT2 123263625 IC50 = 100 nM T08391 CW9BU8 126643886 IC50 = 730 nM T08391 C4BJ8G 126645320 IC50 = 170 nM T08391 CL60VJ 126647240 IC50 = 4400 nM T08391 C1XS8H 126647348 IC50 = 89 nM T08391 CSJ1G7 126647349 IC50 = 19000 nM T08391 C9QCD3 126715362 IC50 = 1770 nM T08391 CNPB25 126715363 IC50 > 30000 nM T08391 CY7US6 126715366 IC50 = 6600 nM T08391 CJS53A 126715367 IC50 = 5010 nM T08391 CX37RN 126715380 IC50 > 15000 nM T08391 C2DQU9 126715387 IC50 > 30000 nM T08391 CH6YP0 126715392 IC50 = 5400 nM T08391 C1QB5R 126715400 IC50 = 1800 nM T08391 CG7YQ2 126715454 IC50 = 322 nM T08391 CO2X6J 126715460 IC50 = 1570 nM T08391 CR9C1G 127030133 IC50 = 150 nM T08391 CU4AJ8 127037981 IC50 = 9620 nM T08391 CA0O1B 127037982 IC50 = 16200 nM T08391 C50NKB 127037983 IC50 > 30000 nM T08391 CF8KQ6 127038326 IC50 = 16200 nM T08391 C5WV8P 127038327 IC50 = 2780 nM T08391 CI8ZB6 127038328 IC50 > 30000 nM T08391 C98DQZ 127038947 IC50 > 17000 nM T08391 CQ4OE5 127039917 IC50 > 22000 nM T08391 CC1XP0 127040339 IC50 = 13900 nM T08391 C8H7JN 127040340 IC50 = 4740 nM T08391 CRQS46 127040341 IC50 > 30000 nM T08391 C3B0AP 127040342 IC50 > 30000 nM T08391 C7KLD9 127040660 IC50 = 10300 nM T08391 C4JF8H 127040661 IC50 = 2270 nM T08391 CC9J7R 127040662 IC50 = 11800 nM T08391 CP1RY4 127040993 IC50 = 2890 nM T08391 C7P5MY 127040994 IC50 = 13100 nM T08391 CB23SC 127041238 IC50 = 14900 nM T08391 CJ7QW5 127041248 IC50 = 9900 nM T08391 C1N6BC 127041249 IC50 = 2700 nM T08391 C5SLH0 127041250 IC50 > 30000 nM T08391 C28YFA 127041251 IC50 > 30000 nM T08391 CIP84Z 127041549 IC50 > 30000 nM T08391 CQP76E 127041550 IC50 > 30000 nM T08391 C3A1VL 127041551 IC50 > 30000 nM T08391 CEJ97D 127041858 IC50 = 1450 nM T08391 C35OPG 127041859 IC50 = 10100 nM T08391 CEN15W 127041860 IC50 = 3040 nM T08391 C4UBE5 127041861 IC50 > 30000 nM T08391 CD1X4L 127045648 IC50 > 1000 nM T08391 CQ76DA 127045649 IC50 > 1000 nM T08391 C4FT6K 127045650 IC50 > 1000 nM T08391 C7Q5YC 127045965 IC50 = 98 nM T08391 C46WVR 127046091 IC50 = 67 nM T08391 C3V5BF 127046092 IC50 = 8 nM T08391 C4SYH9 127046093 IC50 = 21 nM T08391 C5X2VQ 127046094 IC50 = 9 nM T08391 C9YC1K 127046298 IC50 = 78 nM T08391 CQWK04 127046639 IC50 = 732 nM T08391 CZIY10 127046798 IC50 = 531 nM T08391 CX63EC 127046918 IC50 = 184 nM T08391 C6OAX1 127047114 IC50 = 20 nM T08391 CZE85O 127047115 IC50 = 4800 nM T08391 C0R1FI 127047116 IC50 = 1200 nM T08391 CX7LZ6 127047117 IC50 = 908 nM T08391 CAML79 127047118 IC50 > 1000 nM T08391 CCG12W 127047119 IC50 = 155 nM T08391 C2Y1OE 127047142 IC50 = 10 nM T08391 CRYP16 127047143 IC50 = 94 nM T08391 C90NAH 127047271 IC50 = 81 nM T08391 C1UI3Z 127047798 IC50 = 41 nM T08391 CRY8T0 127047799 IC50 = 36 nM T08391 C53OCD 127047800 IC50 = 23 nM T08391 CGA6L4 127047801 IC50 = 6 nM T08391 C26NKY 127047920 IC50 = 17 nM T08391 C19LEF 127047991 IC50 = 97 nM T08391 CS2VY8 127048034 IC50 = 786 nM T08391 CI8Y2P 127048035 IC50 = 475 nM T08391 CB2SE8 127049004 IC50 = 18500 nM T08391 CS6ZO5 127049005 IC50 = 27300 nM T08391 C1PE9L 127050562 IC50 = 3200 nM T08391 CZ5D8C 127050563 IC50 = 29700 nM T08391 CX46RS 127050564 IC50 = 12100 nM T08391 C3LI1J 127050565 IC50 = 3900 nM T08391 CG91WC 127052080 IC50 = 3100 nM T08391 C2LWZ1 129318964 IC50 > 10000 nM T08391 C0FM1R 130196825 IC50 = 170 nM T08391 CZ13WL 130339268 IC50 = 74 nM T08391 CD4NY1 131839645 IC50 = 3.9 nM T08391 C6OXE3 132134663 IC50 = 1.4 nM T08391 CUO0C5 132156633 IC50 > 10000 nM T08391 CV89JM 132231876 IC50 = 3300 nM T08391 CK4FI7 132277003 IC50 > 10000 nM T08391 C5CZA1 132578411 IC50 = 41.9 nM T08391 CDMF97 134130282 IC50 > 100000 nM T08391 C2H6PW 134130554 IC50 = 126 nM T08391 CWF16B 134131331 IC50 = 129 nM T08391 CLV5I3 134131586 IC50 = 50 nM T08391 C5CD9F 134131902 IC50 < 39 nM T08391 CA75NE 134135874 IC50 = 8.9 nM T08391 CR6D9H 134136093 IC50 = 25.7 nM T08391 CQH05W 134136683 IC50 = 18.9 nM T08391 CQ93RF 134136880 IC50 < 39 nM T08391 CG21VI 134136955 IC50 < 39 nM T08391 CDY10C 134137518 IC50 = 136.7 nM T08391 C6VHL4 134137944 IC50 = 324.5 nM T08391 CI0DC7 134138196 IC50 = 6.9 nM T08391 C26PWD 134139689 IC50 = 2.57 nM T08391 C8CP1R 134141659 IC50 = 1.27 nM T08391 CID3G7 134142328 IC50 = 16.6 nM T08391 CFJX74 134142865 IC50 = 1.71 nM T08391 C41ZEF 134143846 IC50 = 7089 nM T08391 C7FXS5 134144592 IC50 = 9 nM T08391 C9Y0KW 134144836 IC50 < 39 nM T08391 CEDU72 134145690 IC50 = 5 nM T08391 C1E2ZW 134145921 IC50 = 4.7 nM T08391 CL9H5I 134146726 IC50 < 39 nM T08391 C8O9SN 134147898 IC50 = 4.3 nM T08391 C48AOM 134150297 IC50 = 10.4 nM T08391 CG9H5W 134150350 IC50 = 2.31 nM T08391 CJX12K 134151832 IC50 = 2.45 nM T08391 CHJ2I6 134152624 IC50 < 39 nM T08391 C96JCY 134153909 IC50 = 30 nM T08391 C4B7IL 134154440 IC50 = 226.1 nM T08391 C8F1BP 134156083 IC50 = 0.97 nM T08391 CCN19D 134157542 IC50 < 39 nM T08391 C1FCZ6 134158025 IC50 = 47 nM T08391 C75NKQ 134537028 IC50 = 1500 nM T08391 CPDT50 134537033 IC50 = 4300 nM T08391 C8CKE5 134537037 IC50 = 1900 nM T08391 C7H8QW 134537039 IC50 = 110 nM T08391 C0ZY5J 134537043 IC50 = 130 nM T08391 CJDM08 134537050 IC50 = 3900 nM T08391 CQ7G4C 134537056 IC50 = 57 nM T08391 CQ1NX6 134537061 IC50 = 27000 nM T08391 C43CFZ 134537067 IC50 = 4800 nM T08391 CELH87 134537071 IC50 = 460 nM T08391 C8DAO7 134537074 IC50 = 18 nM T08391 CQ9OU1 134537081 IC50 = 4500 nM T08391 CH78PN 134537085 IC50 = 1700 nM T08391 CN5P0G 134537092 IC50 = 5900 nM T08391 CHY1S4 134537094 IC50 = 1100 nM T08391 C8L7UN 134537111 IC50 = 110 nM T08391 C42TFN 134537113 IC50 = 690 nM T08391 C58HUF 134537114 IC50 = 1900 nM T08391 C3LRB2 134537119 IC50 = 550 nM T08391 CWU3Z2 134537141 IC50 = 370 nM T08391 CEOW01 134537147 IC50 = 1400 nM T08391 C0T7VN 134537152 IC50 = 2400 nM T08391 CZD72H 134537156 IC50 = 1200 nM T08391 C3HC0S 134537158 IC50 = 240 nM T08391 CTP15L 134537160 IC50 = 3900 nM T08391 C6Z9QY 134537161 IC50 = 430 nM T08391 C9ME6L 134537163 IC50 = 53 nM T08391 CEQ15Z 134537167 IC50 = 4700 nM T08391 C8N6ZF 134537169 IC50 = 3400 nM T08391 CXA39D 134537177 IC50 = 1800 nM T08391 C97OTS 134537185 IC50 = 1300 nM T08391 CHK0V4 134611545 IC50 = 6.6 nM T08391 C20FAE 134611548 IC50 = 83 nM T08391 C51PKU 134611580 IC50 = 5.6 nM T08391 CN75GU 134611727 EC50 = 7710 nM T08391 C80PJI 134611728 IC50 = 48 nM T08391 CFM46L 134812674 IC50 = 366 nM T08391 C2VC5Y 134817793 IC50 = 929 nM T08391 C54FXD 134957362 IC50 > 10000 nM T08391 CVF86X 135125189 IC50 = 3.2 nM T08391 C9MCQ0 135138184 IC50 = 6 nM T08391 C7V2MJ 135142423 IC50 = 2.8 nM T08391 CLET52 135142442 IC50 = 2.1 nM T08391 CU13RW 135142625 IC50 = 7.2 nM T08391 CM7N0J 135142656 IC50 = 22 nM T08391 CG6JI9 135142885 IC50 = 5.6 nM T08391 CQD32R 135143120 IC50 = 9.2 nM T08391 CTJ48K 135524085 IC50 = 3600 nM T08391 CUT1W7 135524168 IC50 = 1300 nM T08391 C7PJ6X 135566704 IC50 > 30000 nM T08391 CI47VJ 135566923 IC50 = 105 nM T08391 CPHG43 135567142 IC50 = 4 nM T08391 C2NRS8 135567293 IC50 = 2.2 nM T08391 C4R1FH 135567294 IC50 = 4.2 nM T08391 CA0R9G 135567295 IC50 = 58.8 nM T08391 CHU3A2 135635724 IC50 = 11000 nM T08391 CPV59N 135685787 Ki > 4000 nM T08391 CRI5F3 135839295 IC50 = 5.4 nM T08391 CH8W7B 135839328 IC50 = 100.8 nM T08391 C29PWN 135886762 IC50 = 3700 nM T08391 CJV08H 135897884 IC50 = 7463 nM T08391 C4K3XL 135897887 IC50 = 551 nM T08391 C93QJC 135897888 IC50 > 10000 nM T08391 CX6JV7 135897894 IC50 = 4410 nM T08391 C5QUL0 135897897 IC50 = 224 nM T08391 CLV7Y8 135897900 IC50 = 589 nM T08391 CFJZ14 135897904 IC50 > 10000 nM T08391 CT2UV5 135897905 IC50 > 10000 nM T08391 CF1PS8 135934877 Ki > 1600 nM T08391 C32BOU 135956049 IC50 = 3 nM T08391 CRU32G 135971388 Ki = 0.8 nM T08391 CTRL59 135976660 Ki = 3500 nM T08391 CJID74 136013449 EC50 = 15800 nM T08391 CHA4N2 136013680 IC50 > 10 nM T08391 C1PCJ3 136042251 IC50 = 830 nM T08391 CHL5Z7 136056540 IC50 = 120 nM T08391 CO0L9T 136056541 IC50 = 190 nM T08391 CLIE18 136056542 IC50 = 1810 nM T08391 CM7V8J 136056543 IC50 > 10000 nM T08391 C64BEV 136056544 IC50 = 83 nM T08391 CP1MX4 136056545 IC50 = 290 nM T08391 C4AR8N 136056546 IC50 = 980 nM T08391 CC10GD 136056547 IC50 = 950 nM T08391 CN1PY3 136056548 IC50 = 184 nM T08391 CI8Y0U 136056549 IC50 > 10000 nM T08391 CY7TJ2 136164051 IC50 = 88 nM T08391 CQ84IZ 136180335 Ki > 4000 nM T08391 CC52HL 136189674 IC50 > 3600 nM T08391 C1YUD0 136219394 IC50 > 10 nM T08391 CIU8W3 136254389 IC50 > 10 nM T08391 C1P6ZW 136263939 IC50 = 0.3 nM T08391 C0R2IL 136901416 IC50 = 6.31 nM T08391 C5JIR2 136987005 IC50 > 100000 nM T08391 CIJ71W 137028350 IC50 = 1300 nM T08391 CS15TL 137028351 IC50 = 2500 nM T08391 CH3M4B 137083628 IC50 > 30000 nM T08391 CJA07O 137083629 IC50 > 30000 nM T08391 C9F8PX 137083630 IC50 > 30000 nM T08391 CE9V4U 137174991 IC50 = 5 nM T08391 CM64UH 137175110 IC50 = 40 nM T08391 C70DIP 137223928 IC50 = 15.9 nM T08391 C9F3KV 137321155 IC50 = 29.6 nM T08391 CJK67W 137321156 IC50 = 3.57 nM T08391 C3Z4AT 137321159 IC50 = 3012 nM T08391 CMY0V2 137321160 IC50 > 6578 nM T08391 CWM9S4 137349398 IC50 = 71 nM T08391 C9I5TJ 137631461 Ki = 900 nM T08391 CAM8K0 137632226 IC50 = 2703 nM T08391 CH9WK1 137632228 IC50 = 11000 nM T08391 C7R2HI 137632648 IC50 = 199 nM T08391 C2I3PY 137633211 IC50 = 658 nM T08391 CJN68H 137633647 IC50 = 538 nM T08391 CF6RH5 137633780 IC50 = 2 nM T08391 C2OC5K 137634207 IC50 = 481 nM T08391 CI1E8V 137634241 IC50 = 236 nM T08391 COE76K 137634328 IC50 = 6.4 nM T08391 C6IU0M 137634461 IC50 = 5 nM T08391 CE4DH3 137635161 IC50 = 770 nM T08391 C6JVG9 137635398 IC50 = 75 nM T08391 CMV38W 137635509 IC50 > 2000 nM T08391 C0VXM3 137635710 Ki = 36 nM T08391 CM73AT 137635759 IC50 = 4670 nM T08391 C63ZFX 137636534 IC50 = 502 nM T08391 CH5SI7 137636771 IC50 = 326 nM T08391 C8FH1S 137637247 IC50 = 200 nM T08391 C8I2NQ 137637573 IC50 = 745 nM T08391 C3RF7B 137638414 IC50 = 1390 nM T08391 CE0ZF8 137638897 IC50 = 5.6 nM T08391 C0J8ZG 137639219 IC50 = 43 nM T08391 C3V4KQ 137641382 IC50 = 219 nM T08391 C50WHR 137641404 IC50 = 377 nM T08391 C2VWE5 137642024 IC50 = 1801 nM T08391 CJ6PU9 137642141 IC50 = 21.2 nM T08391 C0RX1Z 137642404 IC50 = 2.7 nM T08391 CVCM89 137642443 Ki = 3200 nM T08391 CKPB85 137642609 IC50 = 865 nM T08391 C9GDQ6 137642740 IC50 = 2114 nM T08391 CXV15S 137642770 IC50 = 3560 nM T08391 C94ELU 137643208 IC50 > 2000 nM T08391 CO83EQ 137643608 IC50 = 79.6 nM T08391 CQP79B 137643915 IC50 = 788 nM T08391 CGHP09 137645020 IC50 = 0.8 nM T08391 CN34SE 137646319 IC50 > 2000 nM T08391 CI8S5A 137646690 IC50 = 3420 nM T08391 CQYM31 137646825 Ki = 590 nM T08391 CGE91V 137646834 IC50 = 848 nM T08391 CE8SH2 137647292 IC50 = 1270 nM T08391 CUA12V 137647912 Ki = 16 nM T08391 CW6D9H 137648009 IC50 = 1990 nM T08391 C0K5AL 137648444 IC50 = 1200 nM T08391 C9KW2L 137648948 IC50 = 940 nM T08391 CHN7A3 137648975 IC50 = 489 nM T08391 CIB60Q 137649981 IC50 = 7 nM T08391 CF4X3E 137650150 IC50 > 10000 nM T08391 CVHT54 137650515 IC50 = 437 nM T08391 CJQ72A 137650866 IC50 > 10000 nM T08391 CA9K6R 137650880 IC50 = 572 nM T08391 COCF21 137651256 IC50 = 0.5 nM T08391 C3Z7LM 137651481 IC50 = 1.9 nM T08391 CQ27PY 137651710 IC50 = 40.9 nM T08391 CYA52Z 137652173 IC50 = 7 nM T08391 C28QUP 137652864 IC50 > 10000 nM T08391 C6UEB9 137653042 IC50 = 708 nM T08391 CK81UT 137654424 IC50 > 2000 nM T08391 CW6SO7 137654686 IC50 > 3310 nM T08391 CCR5B3 137654793 IC50 = 65 nM T08391 CKM89A 137654900 IC50 = 3.4 nM T08391 C26ONG 137654955 IC50 = 199 nM T08391 CE9OW2 137655154 Ki = 6.6 nM T08391 CVBS03 137656215 IC50 = 0.7 nM T08391 CYWE21 137656346 IC50 = 3.3 nM T08391 C6V3WR 137656619 IC50 = 240 nM T08391 CT1EP3 137656679 IC50 = 17.3 nM T08391 C8VC9A 137657080 IC50 = 7.9 nM T08391 C49GYQ 137658008 IC50 = 244 nM T08391 C59BVH 137658028 IC50 = 2 nM T08391 C6UM5X 137658102 Ki = 370 nM T08391 CO6C8I 137658504 IC50 = 592 nM T08391 CW4CK8 137659037 IC50 = 16 nM T08391 C86KOS 137659382 IC50 = 413 nM T08391 CS61AX 137659496 IC50 > 100000 nM T08391 CR41KW 137660124 IC50 = 0.8 nM T08391 CQ8KF2 137660642 IC50 = 893 nM T08391 CU48TN 137661036 Ki = 150 nM T08391 COMQ54 137661391 IC50 = 939 nM T08391 C5VR2U 137661620 IC50 = 265 nM T08391 CJ52WM 137661888 IC50 = 5437 nM T08391 CO4DP9 137662248 Ki = 14 nM T08391 CU2L5H 138108525 IC50 = 346 nM T08391 C2W0JU 138319690 IC50 > 30000 nM T08391 C28PJZ 138376574 IC50 > 30000 nM T08391 CXV84M 138377596 IC50 = 4 nM T08391 C8X9DR 138584993 IC50 = 109.95 nM T08391 C9NL1M 138585023 IC50 = 0.89 nM T08391 CHX6N7 138585027 IC50 = 3.12 nM T08391 C3RM2Z 138585033 IC50 = 1.07 nM T08391 CBF8S4 138585069 IC50 = 1171 nM T08391 C4O0GC 138585070 IC50 = 17.56 nM T08391 C7KYU3 138585074 IC50 = 140.2 nM T08391 CE5S4Z 138585101 IC50 = 489.65 nM T08391 CM63FA 138585111 IC50 = 14.7 nM T08391 C2U8PZ 138585129 IC50 = 10.55 nM T08391 C0Y2WZ 138585150 IC50 = 72.97 nM T08391 CHMX08 138585151 IC50 = 1.82 nM T08391 CA8N5T 138585156 IC50 = 37.07 nM T08391 CG8TR3 138585164 IC50 = 8.91 nM T08391 C3JR7K 138585184 IC50 > 1000 nM T08391 CQI78V 138585192 IC50 = 37.91 nM T08391 C2UCN9 138605457 IC50 = 14.12 nM T08391 C3RM1U 138605458 IC50 = 229.25 nM T08391 CD4M3W 138605461 IC50 = 63.04 nM T08391 C4VMQ9 138605557 IC50 = 220.8 nM T08391 CQ6R7X 138911330 IC50 = 2700 nM T08391 CI1D9F 139600335 IC50 = 0.7 nM T08391 CI7C4P 140943115 IC50 > 2000 nM T08391 C7U3KH 140943149 IC50 > 2000 nM T08391 C9ZYG8 141366083 IC50 = 5700 nM T08391 C18QDP 141523774 IC50 = 72.3 nM T08391 CD9F4Y 141523776 IC50 = 94.3 nM T08391 C4L6JD 141523781 IC50 = 13.1 nM T08391 CLOI54 141523782 IC50 = 397.4 nM T08391 CDF78Y 141523783 IC50 = 160.3 nM T08391 CSZQ36 141523784 IC50 = 62 nM T08391 CTYQ49 141523785 IC50 = 90.1 nM T08391 C8FC9Y 141531439 IC50 = 469.3 nM T08391 CU51PI 141531440 IC50 = 499 nM T08391 C81RPA 141531442 IC50 = 808.3 nM T08391 CAT46B 141531443 IC50 = 396.2 nM T08391 CS37YV 141531444 IC50 = 1932.5 nM T08391 CEHD51 141728806 IC50 = 12 nM T08391 CCY30N 141728810 IC50 = 22 nM T08391 CLH76T 141728811 IC50 = 20 nM T08391 CQB0U4 141728813 IC50 = 15 nM T08391 CN75MA 141728817 IC50 = 14 nM T08391 CWN43D 141728825 IC50 > 100 nM T08391 C7FW8A 141728827 IC50 = 7 nM T08391 CHS9N0 141728829 IC50 = 21 nM T08391 CN72IC 141728831 IC50 = 10 nM T08391 C7EL5X 141728840 IC50 = 5 nM T08391 C9H8PX 141728841 IC50 = 10 nM T08391 CBV2K5 141728842 IC50 = 36 nM T08391 CZ8J7C 141728843 IC50 = 10 nM T08391 C2HF9A 141728845 IC50 = 61 nM T08391 CBRN42 141728846 IC50 = 46 nM T08391 COEV20 141728855 IC50 > 100 nM T08391 CC03XH 141728860 IC50 = 50 nM T08391 C4RGY1 141728867 IC50 = 46 nM T08391 CNUG79 141728871 IC50 = 30 nM T08391 C65GLX 141728873 IC50 = 5 nM T08391 C9IW0F 141728874 IC50 = 85 nM T08391 C18SJO 141728877 IC50 > 100 nM T08391 CECS13 141753441 IC50 = 1096 nM T08391 C1JR5B 142379949 IC50 = 243 nM T08391 C6C3OH 142744323 IC50 = 156 nM T08391 C45HDA 142744326 IC50 = 96.3 nM T08391 C3SN0Y 142744329 IC50 = 62.7 nM T08391 C2O3RK 142744331 IC50 = 786 nM T08391 C2AWZ6 142744332 IC50 = 210 nM T08391 C4RXO6 142744333 IC50 = 511 nM T08391 CFY17M 142744351 IC50 = 63.6 nM T08391 C5O7KE 142744352 IC50 = 71.8 nM T08391 CM0BL5 142744356 IC50 = 165 nM T08391 C47YDW 142744361 IC50 = 73.5 nM T08391 C2L1ZB 142744367 IC50 = 67.4 nM T08391 CZ6FC4 145362469 IC50 = 450 nM T08391 C6VB3O 145925651 IC50 >= 5000 nM T08391 C2OA9H 145949725 IC50 = 36 nM T08391 CY04PB 145950223 IC50 = 376 nM T08391 CDTW63 145950378 IC50 = 951 nM T08391 CDJ81U 145952312 IC50 = 996 nM T08391 C4BZ0E 145952449 IC50 = 1 nM T08391 C2XP8N 145953005 IC50 > 30000 nM T08391 CA13YG 145953228 IC50 = 16 nM T08391 CN0V3D 145953512 IC50 > 30000 nM T08391 C1OQ3J 145953599 IC50 = 1180 nM T08391 CNS52L 145954024 IC50 = 1030 nM T08391 C4IC5P 145954578 IC50 = 2 nM T08391 CI62ZD 145955000 IC50 = 2 nM T08391 C6QI4B 145955113 IC50 = 8 nM T08391 CRU9F8 145955362 IC50 = 13900 nM T08391 CIP2J9 145955397 IC50 = 357 nM T08391 CZ0K1H 145955759 IC50 = 1 nM T08391 CW2VZ6 145955763 IC50 = 110 nM T08391 CIK4T9 145955799 IC50 = 15 nM T08391 CQ68WS 145956107 IC50 < 3 nM T08391 CZ0B7A 145956262 IC50 = 417 nM T08391 CO6SV3 145957001 IC50 = 6410 nM T08391 C9RH8U 145957804 IC50 = 2 nM T08391 C51ADW 145958260 IC50 = 347 nM T08391 C5XP1C 145958407 IC50 = 3 nM T08391 C3L8IE 145958641 IC50 = 85 nM T08391 C7B2LD 145959014 IC50 = 722 nM T08391 CO05IK 145959360 IC50 = 2 nM T08391 CMCG17 145959462 IC50 = 363 nM T08391 CFC18Z 145960569 IC50 = 18 nM T08391 C2LD5V 145960573 IC50 > 30000 nM T08391 CAGS83 145961653 IC50 = 4 nM T08391 CFY21D 145961655 IC50 = 188 nM T08391 CI9Z7U 145962747 IC50 = 183 nM T08391 CQ86LZ 145963345 IC50 = 765 nM T08391 CPO8J7 145967669 IC50 > 10000 nM T08391 CST35V 145967843 IC50 = 1090 nM T08391 CDNC31 145967951 IC50 > 500 nM T08391 CC3ID7 145968857 IC50 = 3450 nM T08391 C7RF9J 145969339 IC50 = 1420 nM T08391 CWU27Z 145969804 IC50 > 100000 nM T08391 C5VWH3 145970734 IC50 = 46 nM T08391 C63KEL 145970838 IC50 = 3760 nM T08391 CD26ZJ 145970864 IC50 = 1710 nM T08391 C7UG3O 145971121 IC50 = 14100 nM T08391 CEDZ18 145971190 IC50 > 30000 nM T08391 CKPM09 145971514 IC50 = 817 nM T08391 C7K1AJ 145971681 IC50 = 8 nM T08391 CZ85FJ 145972657 IC50 = 1 nM T08391 C7OD0E 145973587 IC50 > 30000 nM T08391 C7TAL5 145979161 IC50 = 41.3 nM T08391 CHVD06 145979212 IC50 > 10000 nM T08391 C7L1IC 145979240 IC50 > 7646 nM T08391 CAJ37B 145979552 IC50 = 1870 nM T08391 CFT50A 145979673 IC50 = 3.4 nM T08391 CE31VG 145979714 IC50 = 1666 nM T08391 C7N8DU 145980127 IC50 = 8623 nM T08391 CWH40Y 145980630 IC50 = 1.8 nM T08391 CX94BD 145980658 IC50 = 9.2 nM T08391 C8AMK1 145980722 IC50 = 1046 nM T08391 C09BPI 145980773 IC50 = 25.6 nM T08391 C81XFH 145980840 IC50 = 4964 nM T08391 C9ZT8Y 145981096 IC50 = 58.3 nM T08391 COG0N1 145981347 IC50 = 239 nM T08391 C85XBC 145981348 IC50 = 470 nM T08391 C2OC6Q 145982084 IC50 = 17 nM T08391 CF8R6Z 145982577 IC50 = 0.96 nM T08391 CHI03D 145982623 IC50 = 0.041 nM T08391 C71AZC 145982856 IC50 = 21 nM T08391 CN4T7U 145982897 IC50 = 2.3 nM T08391 CA7K6C 145983002 IC50 = 40 nM T08391 CEU47V 145983063 IC50 = 867.3 nM T08391 C5VF8P 145983087 IC50 = 508.6 nM T08391 CWS14X 145983289 IC50 = 1397.6 nM T08391 CV28DA 145983327 IC50 = 367.2 nM T08391 CA1LM5 145983443 IC50 = 6.6 nM T08391 CS1GK8 145983460 IC50 = 78.4 nM T08391 CG97VS 145983548 IC50 = 696.8 nM T08391 CML89J 145983552 IC50 = 197.4 nM T08391 CA20KM 145983867 IC50 = 590 nM T08391 CS58RN 145983989 IC50 = 168.4 nM T08391 CJLG54 145984020 IC50 = 0.15 nM T08391 C7THN1 145984160 IC50 = 1118 nM T08391 C30EHD 145984172 IC50 = 2554 nM T08391 CL43AD 145984253 IC50 = 0.04 nM T08391 CODK63 145984420 IC50 = 7.7 nM T08391 CP8J3H 145984569 IC50 = 146.8 nM T08391 C42SJR 145984669 IC50 = 696.8 nM T08391 CLH7K9 145984673 IC50 = 103.5 nM T08391 C67HUC 145984822 IC50 = 590 nM T08391 CXWS04 145984852 IC50 = 3 nM T08391 C2ND4F 145985023 IC50 = 19 nM T08391 CG4U3I 145985120 IC50 = 1420.6 nM T08391 CD1T8G 145985288 IC50 > 1000 nM T08391 C3U9IS 145985565 IC50 = 497.4 nM T08391 C2HXR3 145985769 IC50 = 281.7 nM T08391 CY7X5L 145986106 IC50 = 1947 nM T08391 C03PYD 145986466 IC50 < 1000 nM T08391 C2XPR7 145987380 IC50 = 46 nM T08391 CFH27G 145987566 IC50 = 0.9 nM T08391 CW7V1O 145987719 IC50 > 50000 nM T08391 C8NEY2 145987871 IC50 > 7448 nM T08391 C9ZC0H 145987988 IC50 > 2000 nM T08391 CK6U7Z 145988024 IC50 = 33 nM T08391 C8XBL4 145988088 IC50 = 4.6 nM T08391 C9KJ1A 145988137 IC50 = 97 nM T08391 C0NI8A 145988806 IC50 = 4.3 nM T08391 C9BX4U 145988956 IC50 > 9925 nM T08391 CIVK73 145989244 IC50 > 10000 nM T08391 CI97FM 145989333 IC50 = 2.93 nM T08391 CC8GZ3 145989610 IC50 = 1544 nM T08391 C5I8SR 145989639 IC50 > 10000 nM T08391 CIU9W4 145990027 IC50 > 10000 nM T08391 C3DWZ0 145990496 IC50 > 10000 nM T08391 CTX1A3 145990814 IC50 = 876 nM T08391 CO7F1K 145990990 IC50 = 23 nM T08391 CNG35K 145991262 IC50 > 10000 nM T08391 C0M6LD 145991292 IC50 = 2419 nM T08391 CKGE38 145991618 IC50 = 783 nM T08391 CZ94XS 145991731 IC50 = 18 nM T08391 CJC47L 145992551 IC50 = 95.5 nM T08391 C3RC5J 145992581 IC50 = 2.6 nM T08391 CI8R6P 145992803 IC50 > 10000 nM T08391 CD09RT 145992905 IC50 = 3.1 nM T08391 CG21JZ 145993080 IC50 > 50000 nM T08391 CR2F1Y 145993348 IC50 = 2455 nM T08391 C51DMH 145993445 IC50 > 10000 nM T08391 C51ZNC 145993585 IC50 = 3.9 nM T08391 CF36GI 145993689 IC50 = 109 nM T08391 CSQ7G0 145994254 IC50 = 3.6 nM T08391 C19PRG 145998263 IC50 = 100000 nM T08391 C1S2ER 146025986 IC50 = 2200 nM T08391 CJ8B7I 146185140 IC50 = 48 nM T08391 CHQU21 146185142 IC50 = 26 nM T08391 CS92OU 146185145 IC50 = 119 nM T08391 CXTH86 146185148 IC50 = 35 nM T08391 CP96SV 146185154 IC50 = 461 nM T08391 C71KXB 146185156 IC50 = 16 nM T08391 C9IA1X 146185163 IC50 = 3 nM T08391 CS0OL6 146185170 IC50 = 6 nM T08391 C1IAH7 146185174 IC50 = 27 nM T08391 CXGV39 146185193 IC50 = 37 nM T08391 CZX3B5 146185203 IC50 = 3400 nM T08391 C35CPK 146185546 IC50 = 3049 nM T08391 C5DAO2 149003255 IC50 = 437.1 nM T08391 CZ0LP6 150496562 IC50 = 18 nM T08391 CONR74 154637047 IC50 = 9.3 nM T08391 C7HKA9 154637067 IC50 = 11 nM T08391 CL9P8H 154637078 IC50 = 27 nM T08391 C5T7UA 154701267 IC50 = 24 nM T08391 C7PLT9 155510967 IC50 > 4216 nM T08391 C1WRE2 155511764 IC50 = 2 nM T08391 CR1SE8 155511850 IC50 = 1083 nM T08391 C91YXU 155511860 IC50 = 642.1 nM T08391 CDY5U0 155512704 IC50 = 182 nM T08391 CT9B4M 155512787 IC50 = 437 nM T08391 C2MD1Q 155513187 IC50 > 10000 nM T08391 CM95KR 155513637 IC50 = 396.4 nM T08391 C83ZSG 155514311 IC50 = 160 nM T08391 C7MJY5 155514805 IC50 = 45 nM T08391 CUIO35 155516044 IC50 = 11.5 nM T08391 CD6YR0 155516192 IC50 = 870.4 nM T08391 CTP29J 155516678 IC50 = 2.4 nM T08391 C9VK3I 155517004 IC50 > 50000 nM T08391 C2X8HA 155517088 IC50 > 50000 nM T08391 CE2Q3D 155517448 IC50 = 380 nM T08391 C0E7WS 155518120 IC50 = 692 nM T08391 CDTG10 155518349 IC50 = 5 nM T08391 CQ19HO 155518921 IC50 = 560 nM T08391 CLK4S9 155519594 IC50 = 411 nM T08391 CF0H9V 155520176 IC50 = 503 nM T08391 C0A9LX 155520276 IC50 > 10000 nM T08391 C4YJN9 155520341 IC50 = 77 nM T08391 C1PJC7 155520619 IC50 > 30000 nM T08391 C0YEX7 155521332 IC50 = 370 nM T08391 CLZ08K 155522634 IC50 = 604.7 nM T08391 CXG4L3 155522806 IC50 = 2 nM T08391 CEU10G 155522970 IC50 = 112 nM T08391 C9LUO3 155523352 IC50 = 2500 nM T08391 C7NVQ5 155523535 IC50 = 6.5 nM T08391 C32POG 155523862 IC50 = 57.2 nM T08391 C1HWG6 155524274 IC50 = 102 nM T08391 CU7EQ5 155525897 IC50 = 29.8 nM T08391 CE4FX7 155525956 IC50 = 14.8 nM T08391 C39EGQ 155526165 IC50 = 589.5 nM T08391 CCS24O 155527492 IC50 = 82.1 nM T08391 CK14UT 155528172 IC50 = 2782 nM T08391 CB26JT 155528364 IC50 = 110 nM T08391 CVW07K 155528897 IC50 = 3 nM T08391 CMIC15 155529301 IC50 = 35.4 nM T08391 CL47NH 155529550 IC50 = 1800 nM T08391 CX0B9Q 155530477 IC50 = 5.8 nM T08391 CT9R6V 155530931 IC50 = 65 nM T08391 C67TQL 155530972 IC50 = 194 nM T08391 CRX08F 155531665 IC50 > 30000 nM T08391 CQU09F 155532106 IC50 = 30000 nM T08391 C5V6PY 155532206 IC50 > 2000 nM T08391 C4LE7Q 155532724 IC50 = 30 nM T08391 C75AKY 155533695 IC50 > 2000 nM T08391 CLSV71 155533995 IC50 = 1700 nM T08391 CGH63O 155534464 IC50 = 4 nM T08391 CM0U3I 155534552 IC50 > 1000 nM T08391 C2NPE6 155534808 IC50 = 220 nM T08391 C64FIW 155534972 IC50 = 3148 nM T08391 CE8QW2 155535975 IC50 = 50 nM T08391 C2CG1A 155537016 IC50 > 10000 nM T08391 C06JDH 155537151 IC50 = 190 nM T08391 CMV7B2 155538485 IC50 > 30000 nM T08391 C5GNH8 155538704 IC50 = 2790 nM T08391 C5WB0T 155539358 IC50 = 3540 nM T08391 C03BNT 155539537 IC50 = 3230 nM T08391 C3O6KI 155540160 IC50 = 345 nM T08391 C0D8OL 155540191 IC50 = 7.943 nM T08391 C16MHE 155540242 IC50 > 2000 nM T08391 CBA08W 155540345 IC50 = 820 nM T08391 CP2NY0 155540484 IC50 = 5.012 nM T08391 CF8O5T 155540488 IC50 = 3162.28 nM T08391 C51JNT 155540621 IC50 = 10 nM T08391 C5BTX7 155540994 IC50 = 985.9 nM T08391 C76QBR 155541045 IC50 > 30000 nM T08391 CT1AX5 155541077 IC50 = 7.943 nM T08391 CY8F7S 155541097 IC50 = 538 nM T08391 CH6LV1 155541475 IC50 = 19.95 nM T08391 CS58BA 155541478 IC50 = 1444 nM T08391 CF9AX3 155542099 IC50 = 24 nM T08391 C1B6EK 155542401 IC50 = 25.12 nM T08391 CH59RW 155542578 IC50 = 67 nM T08391 CKL31P 155542961 IC50 = 158.49 nM T08391 CH46TG 155543289 IC50 > 3000 nM T08391 C1QRZ2 155543349 IC50 = 146 nM T08391 CRA21U 155543538 IC50 = 916 nM T08391 CD9Z3W 155544141 IC50 = 2.3 nM T08391 CWSG67 155544202 IC50 = 914.5 nM T08391 CZ3YI6 155544372 IC50 = 583 nM T08391 CTQ63L 155544706 IC50 = 19.95 nM T08391 CP7XE1 155545114 IC50 = 19.95 nM T08391 CFR42U 155545338 IC50 = 158.49 nM T08391 C5BHW8 155546008 IC50 = 18 nM T08391 C5U8HP 155546232 IC50 = 10 nM T08391 CJ8F7V 155546474 IC50 = 6340 nM T08391 CO7ZM2 155546902 IC50 = 13.8 nM T08391 CSI1U9 155547916 IC50 = 260 nM T08391 C0B3RK 155547921 IC50 = 199.53 nM T08391 C3DZU0 155548345 IC50 = 200 nM T08391 C67AYP 155548399 IC50 = 28.8 nM T08391 CPR01A 155549631 IC50 = 126 nM T08391 CI6Y5Z 155549690 IC50 = 7.943 nM T08391 CO6ID4 155550122 IC50 = 43 nM T08391 C10OSG 155550219 IC50 = 190 nM T08391 C3DW8J 155550308 IC50 = 15.85 nM T08391 C31QUW 155550462 IC50 = 25 nM T08391 C6UJS7 155550600 IC50 = 240 nM T08391 C2RQT8 155550913 IC50 > 500 nM T08391 C0DMP2 155551420 IC50 = 2098 nM T08391 CHM8G1 155551600 IC50 = 1970 nM T08391 CX0HL6 155552133 IC50 = 1162.8 nM T08391 C2Q1LR 155552255 IC50 = 2400 nM T08391 CW1UX0 155552333 IC50 = 19.95 nM T08391 CV4NX3 155552736 IC50 = 1540 nM T08391 C62ERW 155552853 IC50 = 79.43 nM T08391 CPB6M8 155553409 IC50 = 1015 nM T08391 C5HQ7X 155553551 IC50 = 57 nM T08391 CADO35 155554376 IC50 = 38 nM T08391 CNTP52 155554413 IC50 = 306 nM T08391 CWLC85 155554605 IC50 = 7.2 nM T08391 CQ6S8E 155554939 IC50 = 19.95 nM T08391 C47MNG 155554972 IC50 > 30000 nM T08391 CP39ZD 155555305 IC50 = 125.89 nM T08391 C28MLB 155555377 IC50 = 15200 nM T08391 C9J4HM 155555486 IC50 = 7851 nM T08391 CTRV23 155555922 IC50 > 30000 nM T08391 CG48UE 155556474 IC50 = 10 nM T08391 C8TYG7 155556520 IC50 > 10000 nM T08391 C59HKP 155557055 IC50 > 3000 nM T08391 CZUT98 155557375 IC50 = 28 nM T08391 CG9E7Z 155557901 IC50 = 23 nM T08391 CHW4O3 155558352 IC50 = 7.943 nM T08391 C7HFI8 155558403 IC50 = 1 nM T08391 C7WND0 155558729 IC50 = 684 nM T08391 C3V5HL 155559143 IC50 = 9.7 nM T08391 C2U5ZM 155559343 IC50 = 25.12 nM T08391 CANJ25 155559746 IC50 = 1000 nM T08391 C46KLS 155559780 IC50 = 45.3 nM T08391 CNK81M 155560413 IC50 = 31.62 nM T08391 C54NQC 155561203 IC50 = 488 nM T08391 C1Z6IL 155561218 IC50 = 350 nM T08391 CRU0K3 155563465 IC50 = 3250 nM T08391 C68TCL 155563799 IC50 = 2043 nM T08391 C8HN2B 155563943 IC50 = 36 nM T08391 C1NM2T 155564180 IC50 = 101 nM T08391 CBQN81 155564466 IC50 > 3000 nM T08391 CZ2NK9 155565077 IC50 = 1995.26 nM T08391 CA0Z1U 155565486 IC50 = 1680 nM T08391 CSNF76 155565806 IC50 = 19.95 nM T08391 CF1X5I 155566525 IC50 = 329 nM T08391 C7S5MC 155566661 IC50 > 3000 nM T08391 CQA46B 155566981 IC50 = 2780 nM T08391 CQ5ZX3 155567095 IC50 = 76600 nM T08391 CSRZ04 155567801 IC50 = 280 nM T08391 CGX28M 155567987 IC50 > 30000 nM T08391 COS7X5 155568028 IC50 = 73.1 nM T08391 COGC41 155568181 IC50 = 8 nM T08391 C0L6UT 155568261 IC50 = 19.95 nM T08391 CR79DJ 155568314 IC50 = 366 nM T08391 CRHE56 155569596 IC50 = 9530 nM T08391 CE50IC 155569626 IC50 = 2000 nM T08391 C3X6WU 155569641 IC50 = 718 nM T08391 C14DIR 16750188 IC50 = 130 nM T08391 C5UI4F 16750189 IC50 = 260 nM T08391 C6JKT9 16750206 IC50 = 230 nM T08391 CYIU14 16750228 IC50 = 24 nM T08391 CX4I6T 16750253 IC50 = 36 nM T08391 CI79TY 16750254 IC50 = 60 nM T08391 CS6UT4 16750288 IC50 = 41 nM T08391 COM3C1 16750290 IC50 = 25 nM T08391 CI67WG 16750292 IC50 = 7 nM T08391 CIGJ63 16750308 IC50 = 77 nM T08391 CL2SY5 16750330 IC50 = 330 nM T08391 CE5P2I 53363072 IC50 = 83 nM T08391 CTV60O 53363073 IC50 = 84 nM T08391 CD74BW 53363074 IC50 = 120 nM T08391 CU3M8P 53363075 IC50 = 150 nM T08391 C07FTA 53363076 IC50 = 220 nM T08391 C9JX2G 53363150 IC50 = 15 nM T08391 CJ04SF 53363151 IC50 = 22 nM T08391 CO7Z2P 53363152 IC50 = 22 nM T08391 C1T2LY 53363154 IC50 = 48 nM T08391 C9GEA7 53363242 IC50 = 96 nM T08391 CA06ID 53363244 IC50 = 35 nM T08391 CTSP38 53363245 IC50 = 44 nM T08391 CM7BZ3 53363246 IC50 = 17 nM T08391 C0QON7 53363337 IC50 = 24 nM T08391 CU76JB 53363338 IC50 = 19 nM T08391 C2PU3M 53364335 IC50 = 1200 nM T08391 C10FXI 53364337 IC50 = 70 nM T08391 C2U9QE 53364338 IC50 = 53 nM T08391 D00ERW 44444843 Ki > 1453 nM T08391 D00HVA 11624601 Ki > 1500 nM T08391 D02BXJ 46864270 IC50 = 536 nM T08391 D02NNT 53232451 IC50 < 1 nM T08391 D03BQI 3794 IC50 > 10000 nM T08391 D04NGS 5330790 IC50 = 2960 nM T08391 D05MHL 44605611 Ki = 0.001 nM T08391 D06HVH 54613583 IC50 > 10000 nM T08391 D07OXC 11650194 IC50 > 25000 nM T08391 D08HFG 24809764 IC50 = 3200 nM T08391 D09HVH 135566652 IC50 > 10 nM T08391 D0D6MH 11617559 IC50 > 13000 nM T08391 D0E0XV 9903786 Ki = 5 nM T08391 D0E5IP 3795 IC50 > 10000 nM T08391 D0E7VO 59627005 IC50 = 68.3 nM T08391 D0GN5Z 5281295 IC50 = 9320 nM T08391 D0H7DQ 6419755 IC50 = 3850 nM T08391 D0I3EY 11492186 IC50 = 1600 nM T08391 D0IR6U 5494425 IC50 = 1 nM T08391 D0J3LR 11634725 Ki > 4000 nM T08391 D0K5UF 72710568 IC50 = 12 nM T08391 D0ME9B 46868971 IC50 > 10 nM T08391 D0OP3D 25099184 Ki = 0.45 nM T08391 D0P6JS 11675054 IC50 > 10000 nM T08391 D0Q3NG 11715520 Ki > 1500 nM T08391 D0R2WK 16038120 IC50 = 1505 nM T08391 D0S7IE 11658882 Ki > 1500 nM T08391 D0US9O 45275255 IC50 < 3 nM T08391 D0V6VQ 53344620 IC50 = 123.6 nM T08391 D0VC0I 5169 IC50 > 100000 nM T65197 C7YS4T 44302558 IC50 = 10000 nM T65197 CF3JU5 44302559 IC50 = 4000 nM T65197 CJ89HD 44302650 IC50 = 85000 nM T65197 CMJH12 44302679 IC50 = 10000 nM T65197 CTD89W 44302692 IC50 = 36000 nM T65197 C3OJ7C 44302695 IC50 = 40000 nM T65197 C0VK8M 44302711 IC50 = 35000 nM T65197 CHE2L6 44302781 IC50 = 10000 nM T65197 CKJ2T6 44302802 IC50 = 1500 nM T65197 C0EC1T 44302803 IC50 = 2000 nM T65197 CP87MZ 44302809 IC50 = 85000 nM T65197 CSN25L 44302825 IC50 = 75000 nM T65197 CHT3Q4 44302858 IC50 = 40000 nM T65197 C54RGJ 44302859 IC50 = 145000 nM T65197 CBGH38 44302864 IC50 = 7000 nM T65197 C5UZY1 44302865 IC50 = 6000 nM T65197 CAIF14 44302873 IC50 = 100000 nM T65197 CL68TP 44302874 IC50 = 1500 nM T65197 CO3GV9 44302893 IC50 = 28000 nM T65197 C3Y7WN 44302894 IC50 = 18000 nM T65197 C1U0JO 44302910 IC50 = 35000 nM T65197 C27FRP 44302937 IC50 = 30000 nM T65197 COIY30 44302942 IC50 = 10000 nM T65197 CI18AN 44303087 IC50 = 42000 nM T65197 CE49GW 44303113 IC50 = 30000 nM T65197 CV9F4Z 44303147 IC50 = 35000 nM T65197 CDCV03 145983254 EC50 = 540 nM T65197 C2S4HG 145983372 EC50 = 42 nM T65197 CICW52 145983477 EC50 = 31 nM T65197 CMRL18 145983483 EC50 = 12 nM T65197 CN8AS4 145984303 EC50 = 240 nM T65197 C49YZK 145984525 EC50 = 540 nM T65197 CNAW82 145985265 EC50 = 31 nM T65197 CQ20OJ 145985501 EC50 = 26 nM T65197 CI70VE 145985981 EC50 = 11 nM T65197 CU8C3V 145986198 EC50 = 540 nM T83011 D01ZSO 4235 Ki = 1080 nM T83011 D03GET 4055 Ki = 400 nM T83011 D04AIT 5280445 IC50 = 59700 nM T83011 D06OMW 3052776 Ki = 7.6 nM T83011 D07UYO 441401 IC50 = 2100 nM T83011 D08KBK 11234049 IC50 = 5700 nM T83011 D09QDP 4380 IC50 = 1690 nM T83011 D0B3HD 2519 IC50 > 50000 nM T83011 D0E7PQ 5311 IC50 > 100000 nM T83011 D0H0HJ 19493 IC50 = 560 nM T83011 D0J2MJ 26758 IC50 = 6.59 nM T83011 D0K8KX 5280343 IC50 = 38660 nM T83011 D0NS6H 3152 IC50 = 15000 nM T83011 D0P9AC 3675 Ki = 94 nM T83011 D0R0UJ 4688 Ki = 20.3 nM T83011 D0S2UG 26757 IC50 = 1.3 nM T83011 D0T1LK 4908 IC50 = 94500 nM T83011 D0T3LF 5826 Ki = 280000 nM T83011 D0TV6I 131682 Ki = 2.29 nM T83011 D00VUI 6199 IC50 > 60000 nM T83011 D07SDQ 969516 Ki = 21500 nM T83011 D0B4VE 10251 IC50 = 2870 nM T83011 D0C3UC 208907 IC50 = 37100 nM T83011 D0F4ZY 5311037 Ki = 27 nM T83011 D0H7PW 638024 IC50 = 483 nM T83011 D0I4ZN 66571643 IC50 > 100000 nM T83011 D0L4FS 5280961 IC50 = 6800 nM T83011 D0U3EP 445154 IC50 = 5010 nM T83011 D0W7LO 9947954 IC50 = 4.1 nM T83011 D00OWF 5280953 Ki = 120800 nM T83011 D02EME 137653313 IC50 = 5900 nM T83011 D02FRR 77844720 IC50 = 1.52 nM T83011 D04AXC 46829776 IC50 = 18800 nM T83011 D06BFA 77844660 IC50 = 123 nM T83011 D06QRW 71307 Ki = 3.9 nM T83011 D08YYW 77844717 IC50 = 2.26 nM T83011 D0AF7J 77844718 Ki = 0.29 nM T83011 D0K2LB 77844666 Ki = 2.39 nM T83011 D0NB7Z 46829772 IC50 = 6900 nM T83011 D0R6RT 137652717 IC50 = 4400 nM T83011 D0U9TR 53262706 IC50 = 253 nM T83011 D0UL2R 77844722 Ki = 0.48 nM T83011 D01LAC 6437850 IC50 = 10 nM T83011 D0IZ1D 44571 IC50 = 23400 nM T83011 CX2C4B 4289 Ki = 32.2 nM T83011 C2ZB4C 5530 IC50 = 2950 nM T83011 CK4N7S 6293 IC50 > 60000 nM T83011 CV6BH8 6809 IC50 = 134000 nM T83011 CI8X6J 6885 IC50 = 28600 nM T83011 CJD54S 7578 Ki = 7240 nM T83011 C1G4XA 8764 Ki = 131000 nM T83011 CP0O8I 9513 IC50 = 761500 nM T83011 CSCE03 9688 IC50 = 7870 nM T83011 CUV23A 10286 IC50 = 54900 nM T83011 C5SRE2 10658 IC50 = 2730 nM T83011 C8H4SX 10724 IC50 = 18600 nM T83011 C5NKT4 15362 Ki = 1000 nM T83011 C0PFU5 21107 IC50 > 1000000 nM T83011 C6IN5F 22860 Ki = 5510 nM T83011 C5IK6F 24383 IC50 = 11700 nM T83011 C3IEL1 26861 IC50 > 100000 nM T83011 C3VL1J 27694 Ki = 29000 nM T83011 C64WMG 52356 IC50 = 2620 nM T83011 C09AHX 68081 IC50 > 60000 nM T83011 CQDJ08 69988 IC50 = 8900 nM T83011 C6V0XN 70385 IC50 = 11810 nM T83011 C6UKD8 74342 IC50 = 1960 nM T83011 CYP9Q7 77135 Ki = 60300 nM T83011 CRXH06 77553 IC50 = 14450 nM T83011 CO7Z4L 77793 IC50 = 27870 nM T83011 CZY6R3 78027 Ki = 97000 nM T83011 CMQ6U7 81528 Ki = 70 nM T83011 CB04TP 83054 Ki = 58100 nM T83011 CQ1RK5 87112 IC50 = 23500 nM T83011 C3P1QX 88562 Ki = 3000 nM T83011 C5HO0S 92892 Ki = 10100 nM T83011 CK1H3L 97662 IC50 > 20000 nM T83011 C5F2TM 98689 IC50 = 1950 nM T83011 C4VE6D 99562 IC50 > 10000 nM T83011 CIF4J3 114679 IC50 = 50000 nM T83011 C7K3SF 120014 IC50 = 45520 nM T83011 C01QZU 127234 IC50 > 100000 nM T83011 C6L0WU 133354 IC50 = 33400 nM T83011 C8W9IH 138472 Ki = 49500 nM T83011 CPO73H 140635 IC50 = 15800 nM T83011 CZ45BJ 147354 IC50 = 3430 nM T83011 CUZN14 156448 Ki = 1900000 nM T83011 C1ND9W 161665 IC50 > 20000 nM T83011 C2QHX7 177014 IC50 > 20000 nM T83011 C1CEJ8 182118 IC50 > 100000 nM T83011 C3KF7H 189206 Ki = 510000 nM T83011 CJ87DC 189208 Ki = 1040000 nM T83011 CF43TE 199605 IC50 = 16.73 nM T83011 CXE58T 217219 IC50 = 38904.51 nM T83011 CW8R2J 223515 Ki = 450 nM T83011 C69FVR 223547 Ki = 10350 nM T83011 CACH74 223561 Ki = 7840 nM T83011 CNL5A0 223570 Ki = 2160 nM T83011 C2C8KI 245226 IC50 = 110 nM T83011 C9R4QN 252037 IC50 = 17720 nM T83011 CY5MJ0 252608 IC50 = 760 nM T83011 C6PDH2 252679 IC50 = 19.5 nM T83011 C3A9FD 255751 IC50 = 500 nM T83011 CDB2W6 267093 Ki = 1000 nM T83011 CBM9H4 275641 IC50 = 9.6 nM T83011 C4PUL2 343657 IC50 = 17600 nM T83011 C5RMJ2 347809 IC50 = 15390 nM T83011 CE8CT9 352026 IC50 = 33200 nM T83011 C69DUA 352028 IC50 = 1860 nM T83011 CLE50D 355690 IC50 = 21590 nM T83011 CS2F1T 371801 IC50 = 2130 nM T83011 CRDH87 379339 IC50 = 10.96 nM T83011 CDE46Q 379340 IC50 = 8.318 nM T83011 C89IEH 379341 IC50 = 130 nM T83011 CK59BP 422521 Ki = 2390 nM T83011 C7HME8 439246 IC50 = 288000 nM T83011 C8N6PO 442186 Ki = 1600000 nM T83011 CK1I4O 466269 IC50 = 49720 nM T83011 CB32AN 473589 IC50 = 550 nM T83011 CMT3P0 480764 IC50 > 100000 nM T83011 C14AWI 499408 Ki = 695000 nM T83011 CNE61X 513102 IC50 = 238.6 nM T83011 CNE01L 513103 IC50 = 58530 nM T83011 CYEV86 513106 IC50 = 7370 nM T83011 C8SR2F 513107 IC50 = 3090295.43 nM T83011 C37CEM 513108 IC50 = 4590 nM T83011 C8WBA4 555203 IC50 = 2238.72 nM T83011 CX8VI4 561354 IC50 = 0.912 nM T83011 CYAZ16 561371 IC50 = 785 nM T83011 C7N6MD 580653 IC50 = 63.2 nM T83011 CP8L0V 599722 IC50 = 3.22 nM T83011 CV36NW 607796 IC50 = 23200 nM T83011 COVU71 613852 Ki = 580000 nM T83011 C0D1XP 616747 IC50 = 50000 nM T83011 C4VIH5 636991 IC50 > 100000 nM T83011 C2IRO1 638256 IC50 = 24090 nM T83011 C0C7MF 641818 IC50 = 471 nM T83011 C4KYW6 649393 IC50 = 13460 nM T83011 CD8KC2 673374 IC50 > 100000 nM T83011 CP91NX 677915 IC50 = 532 nM T83011 CYD46X 680536 IC50 = 257.04 nM T83011 CR9Y7H 680602 IC50 = 3300 nM T83011 CZ7XE1 680623 IC50 = 497 nM T83011 C5QIK2 682145 IC50 = 6390 nM T83011 CPIT91 682187 IC50 = 10460 nM T83011 C8WL2S 688763 IC50 = 18070 nM T83011 CDE9V2 689424 IC50 = 4500 nM T83011 C5O0TJ 690158 IC50 = 5650 nM T83011 CP91KB 691961 IC50 = 29420 nM T83011 CM51LR 692546 IC50 > 10000 nM T83011 CUHY04 692606 IC50 = 5210 nM T83011 C46VZA 692702 IC50 = 666 nM T83011 C61FYO 693313 IC50 = 2530 nM T83011 CQV73I 694612 IC50 = 67 nM T83011 CT9R3F 694735 IC50 = 4890 nM T83011 CC40ZA 711807 IC50 = 348 nM T83011 CU4IZ0 724176 IC50 = 650 nM T83011 CLH57V 724182 IC50 = 35400 nM T83011 C19WBZ 724184 IC50 = 640 nM T83011 CJ01NQ 724189 IC50 = 2960 nM T83011 CVJ15O 724191 IC50 = 13740 nM T83011 CQ59DC 724193 IC50 = 22450 nM T83011 C3YOJ2 724194 IC50 = 18270 nM T83011 C2NVT7 724195 IC50 = 380 nM T83011 CIS57F 724196 IC50 = 700 nM T83011 C9NYF1 728520 IC50 = 1.585 nM T83011 C3SI7X 731731 IC50 = 7.01 nM T83011 C6SQ9Y 735483 IC50 = 930 nM T83011 CL7HM5 736681 IC50 = 6700 nM T83011 C8J0PG 737170 IC50 = 2820 nM T83011 C6UPH7 740329 IC50 = 9.03 nM T83011 C69QTF 745287 IC50 = 820 nM T83011 C32QRF 746682 IC50 = 21630 nM T83011 C54GJN 747648 IC50 = 95.5 nM T83011 CV6ZP4 747794 IC50 = 39110 nM T83011 CB25MU 748172 IC50 = 2010 nM T83011 CC5R0A 748253 IC50 = 200 nM T83011 C1E9FW 748372 IC50 = 250 nM T83011 COM0W3 748376 IC50 = 50030 nM T83011 CL9GS4 764149 IC50 = 5280 nM T83011 CSB8C7 767956 IC50 = 5.95 nM T83011 CV7CU9 771016 IC50 = 58380 nM T83011 CTON48 780558 IC50 = 18.9 nM T83011 CTRO75 781371 IC50 = 4180 nM T83011 CV9KO3 785047 IC50 = 47.24 nM T83011 C2U0LO 794222 IC50 = 3180 nM T83011 C27LMJ 797192 IC50 = 860 nM T83011 C5PDK8 802516 IC50 = 1950 nM T83011 CR98SI 804903 IC50 = 19.43 nM T83011 CAKL20 807313 IC50 = 0.912 nM T83011 CDU38G 834420 Ki = 1073 nM T83011 CK2Z1F 852572 IC50 = 1580 nM T83011 CGCD65 871734 IC50 = 1130 nM T83011 CF89IZ 872422 IC50 = 1290 nM T83011 CYVA98 874919 IC50 = 447 nM T83011 C72NHE 877852 IC50 = 1410 nM T83011 COI0G4 882597 IC50 = 1.38 nM T83011 C3XY5A 882744 IC50 = 2.138 nM T83011 CLD6K7 882800 IC50 = 1.072 nM T83011 CSX7H6 882845 IC50 = 6.48 nM T83011 CBG9N4 883299 IC50 = 1.202 nM T83011 C53RQI 883300 IC50 = 1.549 nM T83011 C6GM0Z 886539 IC50 = 0.9 nM T83011 COUL71 891711 IC50 = 1210 nM T83011 C8T7IX 894515 IC50 = 3.236 nM T83011 CQ4I9A 894713 IC50 = 2620 nM T83011 CIN30B 894965 IC50 = 16.5 nM T83011 C3ST1B 895155 IC50 = 114 nM T83011 C02WCM 895200 IC50 = 10.52 nM T83011 CC8IJ5 895343 IC50 = 75.4 nM T83011 C6C5JT 904559 IC50 = 1.66 nM T83011 C02JTM 915272 IC50 = 3090 nM T83011 C0MS5E 927669 IC50 > 50000 nM T83011 COY2I6 939812 IC50 = 1.122 nM T83011 CZFU46 958268 IC50 = 105 nM T83011 CUMA52 965710 IC50 = 11.48 nM T83011 CIT3L2 1016023 IC50 = 30590 nM T83011 C4YAE7 1037029 IC50 = 199 nM T83011 CLV13S 1111873 IC50 = 20170 nM T83011 C5S2LQ 1178193 IC50 = 11550 nM T83011 CKFO95 1201119 IC50 = 6070 nM T83011 C47DQB 1211950 IC50 = 880 nM T83011 C82HEY 1241457 IC50 = 2570 nM T83011 C7EGD5 1249836 IC50 = 82 nM T83011 CA84HD 1251882 IC50 = 192 nM T83011 CDVS56 1268920 IC50 = 2490 nM T83011 C9G1NF 1269411 IC50 = 1020 nM T83011 CF7GZ3 1272788 Ki = 2730 nM T83011 CR12NY 1327377 IC50 = 22800 nM T83011 CA9U8F 1332620 IC50 = 104 nM T83011 C0IHA6 1345219 IC50 = 11000 nM T83011 CBW19M 1383560 IC50 = 22000 nM T83011 CED0S4 1416314 IC50 = 604300 nM T83011 C4AR3X 1494342 IC50 = 190 nM T83011 CH70DU 1504749 IC50 = 3800 nM T83011 C4M8RY 1505193 IC50 = 380 nM T83011 C8RV0X 1505221 IC50 = 500 nM T83011 CM80QJ 1509337 IC50 = 100 nM T83011 CENL04 1523065 IC50 = 242 nM T83011 C9TR4H 1523287 IC50 = 10060 nM T83011 C1SH3T 1548910 IC50 = 61000 nM T83011 C8U4BF 1550573 IC50 = 105.51 nM T83011 CXS98U 1551716 IC50 = 2940 nM T83011 CL9UE7 1641788 IC50 = 228 nM T83011 CM02NF 1712168 IC50 = 36480 nM T83011 COB92M 1730869 IC50 = 27500 nM T83011 CBR10Z 1773356 IC50 = 42130 nM T83011 C2AH4U 1778270 IC50 = 64170 nM T83011 CH94OA 1815444 IC50 = 54.77 nM T83011 CQR67C 1909002 Ki = 15150 nM T83011 CW4G6A 1929998 IC50 = 800 nM T83011 C9P2SG 2054475 IC50 = 15400 nM T83011 CZJ21Q 2195073 IC50 = 85.6 nM T83011 CQSP80 2237121 IC50 > 100000 nM T83011 C82KZO 2263916 IC50 = 46070 nM T83011 C6IU4T 2296540 IC50 = 379 nM T83011 CMW1F0 2302856 IC50 = 5000 nM T83011 C05ZWH 2305452 IC50 = 154.23 nM T83011 C73JAP 2305454 IC50 = 1130 nM T83011 C3GPH4 2313594 IC50 = 58.9 nM T83011 CM5XN1 2329351 IC50 = 27000 nM T83011 CEVF10 2455077 IC50 = 247.51 nM T83011 CF81QZ 2629406 IC50 = 0.5 nM T83011 CJXT18 2697319 IC50 = 20892961.31 nM T83011 CQ5W4K 2697325 IC50 = 478630.09 nM T83011 CEQ4V8 2723716 IC50 = 2500 nM T83011 CB1H8U 2728598 IC50 = 68.78 nM T83011 CKA6N4 2728599 IC50 = 65.48 nM T83011 CO3JT6 2728600 IC50 = 10.26 nM T83011 C61MIZ 2737276 IC50 = 12.9 nM T83011 C9XF5A 2756638 IC50 = 2730 nM T83011 C0DSF4 2758968 IC50 = 83.1 nM T83011 CN6Z0G 2758969 IC50 = 1060 nM T83011 C3JSD1 2758970 IC50 = 580 nM T83011 CC2S9E 2759808 IC50 = 1530 nM T83011 C0KB6G 2765447 IC50 = 14.79 nM T83011 CUQR43 2767324 IC50 = 269.15 nM T83011 CCRV24 2767328 IC50 = 8.128 nM T83011 CR84JM 2767331 IC50 = 4.571 nM T83011 CVKF21 2769183 IC50 = 602.56 nM T83011 C9AH7R 2774040 IC50 = 201000 nM T83011 CXDE69 2787564 IC50 = 1.122 nM T83011 CCH4L0 2798381 IC50 = 7900 nM T83011 CUNL56 2801340 IC50 = 96.5 nM T83011 CNP4S1 2806094 IC50 > 100000 nM T83011 CANM16 2827498 IC50 = 921 nM T83011 CLZS72 2834140 IC50 = 5.623 nM T83011 CMJ7R6 2911886 IC50 = 48310 nM T83011 CV1Y6Z 3018343 Ki = 1940000 nM T83011 C0E7TW 3035046 IC50 > 200000 nM T83011 CBR5K8 3035812 IC50 = 2.2 nM T83011 C2XP0H 3052775 IC50 = 14 nM T83011 C3US8W 3076090 IC50 = 2 nM T83011 C4DCJ7 3082143 Ki = 21000 nM T83011 CKD72T 3083848 IC50 = 5440 nM T83011 C0OA8F 3107378 IC50 = 66640 nM T83011 CI34YK 3121217 IC50 = 1.778 nM T83011 CC48UQ 3162481 IC50 = 10000 nM T83011 C2GE9F 3162506 IC50 = 4960 nM T83011 C6IPM8 3391493 IC50 = 40000 nM T83011 C8PH2T 3417338 IC50 = 56000 nM T83011 CX7T5S 3517936 IC50 > 100000 nM T83011 C90THR 3553261 IC50 > 100000 nM T83011 C5DV0S 3596769 IC50 = 530 nM T83011 CCW40J 3670544 IC50 = 251.19 nM T83011 CW6J9Q 3684469 IC50 = 74700 nM T83011 CX0AD8 3778700 IC50 = 2910 nM T83011 C74MFV 3788436 IC50 = 204.17 nM T83011 CJ80EG 3822321 IC50 = 21550 nM T83011 CR9Y4X 3928946 IC50 = 4520 nM T83011 CB49EF 3988576 IC50 = 7960 nM T83011 CF27HP 4082687 IC50 = 23840 nM T83011 CH8RB9 4117727 IC50 = 49960 nM T83011 COQ27R 4149109 IC50 = 460 nM T83011 C18AYX 4313470 Ki = 5300 nM T83011 COJV81 4521898 IC50 = 57.37 nM T83011 C70WJL 4679494 IC50 = 66400 nM T83011 CFQ3J7 4779843 IC50 = 60 nM T83011 CR9K6W 4914973 IC50 = 800 nM T83011 C0X8GM 4914974 IC50 = 4680 nM T83011 CT6GY3 5169444 IC50 = 8050 nM T83011 CS3FA0 5200296 IC50 = 102 nM T83011 C84CKE 5200299 IC50 = 311 nM T83011 C28VXZ 5200300 IC50 = 77.1 nM T83011 C80PSO 5200303 IC50 = 86.3 nM T83011 CX7S2M 5200304 IC50 = 56.9 nM T83011 C9LWZ2 5270542 IC50 = 1100 nM T83011 C3M1CE 5270587 IC50 = 69360 nM T83011 CNZ73E 5280567 IC50 = 80410 nM T83011 CWE84I 5281233 IC50 = 128000 nM T83011 CL1MR9 5281254 Ki = 510 nM T83011 CE5SI3 5281725 IC50 = 3620 nM T83011 C5LGJ1 5282362 IC50 = 182 nM T83011 CLE8F3 5302715 IC50 = 54 nM T83011 CQ7TV2 5314262 IC50 = 3690 nM T83011 CPRI38 5320318 IC50 > 60000 nM T83011 CNA80W 5337609 Ki = 13900 nM T83011 CXCI17 5345068 IC50 = 2450 nM T83011 C9D5NA 5346030 IC50 = 1396 nM T83011 CK1V4C 5346482 IC50 = 500 nM T83011 CXKD41 5348419 IC50 = 624 nM T83011 C7XKQ6 5354125 Ki = 1900000 nM T83011 CPW0G3 5354554 IC50 = 69 nM T83011 CW6IE0 5356384 IC50 > 10000 nM T83011 CH73ZU 5356597 IC50 = 71320 nM T83011 C8ZJ2Q 5357659 Ki = 5550 nM T83011 C7EZA1 5368282 IC50 = 85 nM T83011 CDMP72 5370638 Ki = 35 nM T83011 C7FCX1 5370710 IC50 = 33200 nM T83011 CI1V0M 5372946 IC50 = 160 nM T83011 C4S1UA 5375423 Ki = 2470 nM T83011 CS2VC6 5377023 IC50 = 529 nM T83011 CM3T9J 5377817 IC50 > 10000 nM T83011 C4T1CZ 5388521 IC50 = 31 nM T83011 C57ZGH 5458879 EC50 = 1200 nM T83011 C8QP4J 5467625 IC50 = 305 nM T83011 CCUM24 5467627 IC50 = 99 nM T83011 C7U5IY 5473688 Ki = 1330000 nM T83011 CP9Z3C 5646441 IC50 = 1160 nM T83011 CLC01O 5708964 IC50 = 667.89 nM T83011 CME0C2 5709307 IC50 = 7670 nM T83011 C1QUA7 5711036 IC50 > 10000 nM T83011 CRQ3P9 5711038 IC50 = 1430 nM T83011 C1T4AF 5712162 IC50 = 31 nM T83011 C26HRP 5717651 IC50 = 924 nM T83011 C8A3JH 5717653 IC50 = 619 nM T83011 C6SR2J 5718033 IC50 = 707 nM T83011 C7IZJ1 5723719 IC50 = 16 nM T83011 CKN25F 5727970 IC50 = 1530 nM T83011 CZ79RX 5728224 Ki = 14900 nM T83011 CM7V8F 5729327 Ki = 27000 nM T83011 CVM37E 5731408 IC50 = 3200 nM T83011 CCM41G 5780273 Ki = 7700 nM T83011 CCW54K 5783530 IC50 = 12440 nM T83011 CW0M9V 5784792 IC50 = 419 nM T83011 CU1I8E 5815007 IC50 = 310 nM T83011 C2F4QH 5820198 IC50 = 2290 nM T83011 C7LKC3 5822497 IC50 = 4.4 nM T83011 C7TOI9 5863209 IC50 = 793 nM T83011 CS93TJ 5903767 IC50 = 450 nM T83011 CE59LJ 5908055 Ki = 7220 nM T83011 CK0M4A 5910585 IC50 = 144.54 nM T83011 CJS0P7 5945471 IC50 = 4890 nM T83011 CFN9G8 5989034 IC50 = 56 nM T83011 C5V4SY 6093310 Ki = 2300000 nM T83011 C73HMS 6106285 Ki = 7000 nM T83011 CL9Z1S 6110591 Ki = 4220 nM T83011 C31OYT 6163838 Ki = 2550 nM T83011 CO0IJ3 6212978 IC50 = 4490 nM T83011 CYX45A 6213016 IC50 = 57 nM T83011 CCN49Q 6364799 IC50 = 478630.09 nM T83011 CLR14W 6364800 IC50 = 181.45 nM T83011 CT8N5B 6370756 IC50 = 10510 nM T83011 C49LEJ 6404472 IC50 = 8.511 nM T83011 CAS82I 6409776 IC50 = 5.012 nM T83011 C40RHI 6421573 IC50 = 6536800 nM T83011 CFWP52 6433444 IC50 > 10000 nM T83011 C1N0KP 6436743 IC50 > 10000 nM T83011 CL26DC 6443328 Ki = 380000 nM T83011 C2VZ3C 6443329 Ki = 690000 nM T83011 CYXP79 6449266 IC50 = 104.34 nM T83011 CGOC05 6455277 IC50 = 513 nM T83011 C1VU0Y 6461059 IC50 = 1550 nM T83011 C6BFA8 6461322 IC50 = 228.6 nM T83011 CRDF19 6474563 IC50 > 10000 nM T83011 C2LS0C 6479236 IC50 = 55.37 nM T83011 CDK5A4 6479237 IC50 = 31.82 nM T83011 CM1IN3 6479238 IC50 = 13.03 nM T83011 CKO7Y8 6479239 IC50 = 1570 nM T83011 C75UNJ 6524131 IC50 = 8.51 nM T83011 CGHV31 6864775 IC50 > 10000 nM T83011 CNL1X8 6873295 IC50 > 10000 nM T83011 CUJA07 6896171 IC50 > 10000 nM T83011 C5L8EP 7214067 IC50 > 10000 nM T83011 CM91LR 7559290 IC50 = 7610 nM T83011 CI4NS5 7695078 IC50 > 10000 nM T83011 C58LDF 7728944 IC50 > 10000 nM T83011 COS56D 7946925 IC50 = 133 nM T83011 C60IRP 8438344 IC50 = 910 nM T83011 C0HDR2 8443698 IC50 = 13 nM T83011 C6I0XF 8446625 IC50 = 470 nM T83011 C4P2UQ 8607850 IC50 = 1055 nM T83011 CSW24U 8744495 IC50 = 223 nM T83011 C36XCB 8861814 IC50 = 1310 nM T83011 C95JLG 9412345 IC50 = 283 nM T83011 C18OMT 9413726 IC50 = 580 nM T83011 CQ8IR0 9593639 IC50 = 2220 nM T83011 CB41FJ 9601017 Ki = 120 nM T83011 C8I7XN 9609596 IC50 = 3060 nM T83011 CF4A5O 9637488 IC50 = 3050 nM T83011 CUFX46 9685369 IC50 = 2760 nM T83011 C79LKI 9737735 IC50 = 3840 nM T83011 CB9IF4 9737737 IC50 = 944 nM T83011 CV7W8X 9737770 IC50 = 810 nM T83011 CZ72CK 9799696 IC50 = 47 nM T83011 CVSU04 9817917 IC50 = 60000 nM T83011 CK7ZU5 9837722 IC50 = 86.4 nM T83011 C03JZN 9838864 IC50 = 3884 nM T83011 CFRO05 9904206 Ki = 221.6 nM T83011 C4N1IG 9971058 IC50 = 33.11 nM T83011 CW9X2A 9975046 IC50 = 1288.25 nM T83011 CQ38WI 9975414 IC50 = 128.82 nM T83011 CYO48N 9995644 IC50 = 28.18 nM T83011 CW9T3A 10064939 IC50 = 588.84 nM T83011 C94RLT 10083342 IC50 = 2691.53 nM T83011 CC7OQ6 10086160 IC50 = 26.3 nM T83011 C7IEF9 10095474 IC50 = 2390 nM T83011 CRYQ79 10107929 IC50 = 26.3 nM T83011 C62ZIW 10176672 IC50 = 200 nM T83011 C3PEH7 10246762 IC50 = 5.9 nM T83011 CNPO06 10265999 IC50 = 31.62 nM T83011 CRL70U 10266501 IC50 = 1580 nM T83011 CD7H4C 10314028 IC50 = 0.014 nM T83011 C65QLI 10331501 IC50 > 100000 nM T83011 CCW21R 10334013 IC50 = 117.49 nM T83011 CHZX23 10336709 IC50 = 1080 nM T83011 C7X8OB 10344711 IC50 > 100000 nM T83011 C0LV3E 10357601 IC50 = 524.81 nM T83011 CRF71V 10376837 IC50 = 120 nM T83011 CC3D0F 10378713 IC50 = 42.66 nM T83011 CU5I8C 10379207 IC50 = 711.23 nM T83011 C25WON 10382902 IC50 = 1500 nM T83011 C5ND4S 10403008 IC50 = 6.31 nM T83011 CU2KJ1 10404089 IC50 = 5.37 nM T83011 CJ1H7P 10423365 IC50 = 758.58 nM T83011 CBV6N7 10423722 IC50 = 15.32 nM T83011 CCS6V5 10424451 IC50 = 190.55 nM T83011 C8MA6I 10442609 IC50 > 50000 nM T83011 C0P5WH 10449040 IC50 = 169.82 nM T83011 CZLC86 10468459 IC50 = 2951.21 nM T83011 CN0PA5 10469356 IC50 = 42.66 nM T83011 CG9Z3B 10470997 IC50 = 4.25 nM T83011 C8SFX5 10517814 IC50 = 8.71 nM T83011 C0LAO1 10520909 IC50 = 7.943 nM T83011 CR9SE7 10540319 IC50 = 5.1 nM T83011 CDT28L 10586897 IC50 = 53 nM T83011 C0WH8G 10594917 IC50 = 3.631 nM T83011 CA51UC 10633774 IC50 = 15210 nM T83011 CG65YU 10666829 IC50 = 1.622 nM T83011 CFA2E3 10682241 IC50 = 63 nM T83011 C8YO4I 10682287 Ki = 19 nM T83011 CYV29T 10682625 IC50 = 51 nM T83011 C5W7OY 10685346 IC50 = 125.89 nM T83011 CW67NI 10705194 IC50 = 24 nM T83011 C2SDN4 10732696 IC50 = 3.89 nM T83011 CBO1H0 10826534 IC50 = 1.38 nM T83011 C0OW2P 10850658 IC50 = 860.46 nM T83011 C79PFH 10855817 IC50 = 78860 nM T83011 C7RD3K 10872091 IC50 = 218 nM T83011 C3EHA8 10879393 IC50 = 4280 nM T83011 CU4FD9 10883954 Ki = 60220 nM T83011 C5E8IT 10905291 IC50 = 92000 nM T83011 C7DO5I 10921069 IC50 = 24000 nM T83011 CLK8M1 10970782 IC50 = 624 nM T83011 CPH2B5 10981956 Ki = 69900 nM T83011 C8NS7W 11008446 IC50 > 50000 nM T83011 C3OBZ4 11013275 IC50 = 240000 nM T83011 C5OA1U 11055762 IC50 = 12120 nM T83011 C7I2PD 11075734 IC50 = 50200 nM T83011 CTOC87 11077623 IC50 = 199 nM T83011 CCPK75 11131758 IC50 = 22000 nM T83011 CA3OV1 11205967 IC50 = 13000 nM T83011 CQY25S 11205968 IC50 = 24000 nM T83011 CJD31L 11206576 Ki = 23900 nM T83011 CRC94Z 11217911 IC50 = 6700 nM T83011 CKEG43 11217912 IC50 = 30000 nM T83011 CU9RL6 11219387 Ki = 700000 nM T83011 CMJ81Y 11231451 Ki = 1240 nM T83011 CYL3G8 11252448 IC50 = 3.6 nM T83011 CVR53M 11276756 IC50 = 167 nM T83011 C9Q4IK 11288016 IC50 = 300 nM T83011 CH5D6X 11324053 Ki = 100000 nM T83011 C9T7SG 11333223 Ki = 15000 nM T83011 CYR01F 11333500 Ki = 36000 nM T83011 C8DK6A 11335051 Ki = 520000 nM T83011 C2RJ0V 11335598 Ki = 400000 nM T83011 CLF08H 11355798 IC50 = 38018.94 nM T83011 CI9ST4 11382228 IC50 = 630.96 nM T83011 CKNY71 11414870 Ki = 410000 nM T83011 CN6M2D 11425653 Ki = 500000 nM T83011 CW6TH3 11492515 IC50 = 140000 nM T83011 C5MOH8 11506668 IC50 = 81000 nM T83011 C2BV6C 11508380 IC50 = 11000 nM T83011 CYH39X 11529216 IC50 = 38000 nM T83011 C0FWJ4 11544612 IC50 = 580 nM T83011 CI75BL 11559017 IC50 = 471 nM T83011 CSGK12 11580635 IC50 = 25000 nM T83011 C03FJS 11580776 Ki = 6.88 nM T83011 CXU5I3 11616886 Ki = 100 nM T83011 C2D7FW 11644221 IC50 = 24500 nM T83011 C6O9WD 11658488 IC50 = 650 nM T83011 C92VMW 11673215 IC50 = 88000 nM T83011 CS28CV 11674943 IC50 = 860 nM T83011 C7E9FY 11687666 IC50 = 32480 nM T83011 CD57XZ 11695291 IC50 = 2840 nM T83011 C3WY1J 11702056 IC50 = 305 nM T83011 CQ0VL1 11708681 IC50 = 0.318 nM T83011 CV9R5X 11715359 IC50 = 90000 nM T83011 CQ9JE1 11716117 IC50 = 109 nM T83011 C5V9SU 11747578 IC50 = 75.84 nM T83011 C0E3QZ 11957673 IC50 = 33 nM T83011 CDH46N 11964510 IC50 = 19 nM T83011 C4ATG6 12070966 IC50 > 100000 nM T83011 C6KB9J 12070967 IC50 > 100000 nM T83011 CMW6C0 12142409 Ki = 4270 nM T83011 C2UYL7 12147097 IC50 = 5623.41 nM T83011 C0WYK2 12180960 IC50 = 12300 nM T83011 CL43NJ 12194782 IC50 = 9.2 nM T83011 CM13FC 12200770 IC50 > 1000000 nM T83011 CHXY39 12251868 IC50 = 1330 nM T83011 CO0B3Y 12317147 Ki = 76000 nM T83011 C60LTR 12341471 IC50 = 5160 nM T83011 CTMH07 12370465 IC50 = 33 nM T83011 CET0B9 12536095 IC50 > 100000 nM T83011 C8XI6U 12558853 IC50 = 283.75 nM T83011 CN1I4H 12615313 IC50 = 986 nM T83011 CL19DT 12622120 IC50 = 1905.46 nM T83011 C2OM1D 12654835 IC50 = 70.7 nM T83011 C01ZKC 12743534 IC50 = 11200 nM T83011 C9BKA2 12822089 IC50 > 10000 nM T83011 CL12FG 12887493 IC50 = 31500 nM T83011 C3HIS0 12899541 IC50 = 21800 nM T83011 CO3FX6 13004209 IC50 = 1540 nM T83011 CW31OY 13067328 IC50 = 7 nM T83011 CX1I4T 13067331 IC50 = 33 nM T83011 CFJW72 13108121 IC50 = 18000 nM T83011 C9RH7B 13108122 IC50 = 20300 nM T83011 CY6W5B 13147660 IC50 > 100000 nM T83011 C4CL7K 13212930 Ki = 6200000 nM T83011 C4ARU8 13309301 IC50 = 15.85 nM T83011 CX1BH2 13309305 IC50 = 199.53 nM T83011 C16ULJ 13340059 IC50 = 58.2 nM T83011 C9G6FX 13340060 IC50 = 77.8 nM T83011 CN8Y5U 13340061 IC50 = 21.5 nM T83011 CZ20KX 13441539 IC50 = 0.3085 nM T83011 CSY7V3 13560856 Ki = 129000 nM T83011 C9NHV7 13925346 IC50 = 1184400 nM T83011 CR1GI7 14079439 IC50 = 1060 nM T83011 C2RE9H 14101461 IC50 = 6370 nM T83011 C7BPR5 14101462 IC50 = 13300 nM T83011 CA93TP 14248936 IC50 = 10730 nM T83011 C65XEY 14364356 IC50 > 100000 nM T83011 C8R0DB 14364358 IC50 > 100000 nM T83011 C2AM4B 14364359 IC50 > 50000 nM T83011 CC0PF9 14493789 IC50 = 6490 nM T83011 C6BXJ3 14521594 IC50 = 2.73 nM T83011 CL8CJ0 14570343 IC50 = 2.884 nM T83011 CHS1K3 14669096 IC50 = 1130 nM T83011 CTW86O 14686301 IC50 = 113.21 nM T83011 CAL70P 14686305 IC50 = 45.36 nM T83011 C3H1UG 14737145 IC50 = 3350 nM T83011 CVAM34 14798396 IC50 = 2.344 nM T83011 CL54PD 14798397 IC50 = 1.413 nM T83011 C17ZIC 14798399 IC50 = 4.266 nM T83011 CBZ43L 14807789 IC50 = 38500 nM T83011 CEH9F5 14807793 IC50 > 50000 nM T83011 CJZ87V 14810157 Ki = 513 nM T83011 C6GH0X 14953522 IC50 = 4.4 nM T83011 CTHB49 14953546 IC50 = 8 nM T83011 C8MS7V 14953547 IC50 = 16 nM T83011 C2J8SV 14956421 Ki = 805 nM T83011 C2GJQ3 14956422 Ki = 1800 nM T83011 CCW67A 14956425 IC50 = 39370 nM T83011 CB71PU 14956426 IC50 = 12840 nM T83011 CB4J3X 14985618 IC50 = 4200 nM T83011 CL2I1Y 15184833 IC50 = 33380 nM T83011 CUA6O8 15193131 IC50 = 340 nM T83011 C7Y2EW 15193139 IC50 = 1170 nM T83011 CNX0G2 15234950 Ki = 15000 nM T83011 CHV17I 15324420 Ki = 1880 nM T83011 CN95UR 15370086 IC50 = 17780 nM T83011 CAY8U5 15480987 IC50 = 67.9 nM T83011 C9A1WR 15484393 IC50 = 8.61 nM T83011 CNEI48 15521042 IC50 = 66400 nM T83011 CF6BU2 15569251 IC50 = 7.9 nM T83011 CB09CW 15609636 IC50 = 97.47 nM T83011 CFGD90 15609637 IC50 = 44.18 nM T83011 CB36PW 15634400 IC50 > 100000 nM T83011 C8FSV7 15953790 IC50 = 57 nM T83011 CJV02O 15953792 IC50 = 64200 nM T83011 C21GMP 16099924 Ki = 3670 nM T83011 C0S3XE 16345405 IC50 = 8230 nM T83011 C40MHI 16444239 IC50 = 17440 nM T83011 CASK57 16584098 IC50 = 7.98 nM T83011 C1OP9D 16787761 Ki = 663 nM T83011 C04JHC 16792980 Ki = 44 nM T83011 CXM83Z 17163667 Ki = 5.48 nM T83011 C6X9OR 17165093 Ki = 1459 nM T83011 C6G9JN 17167188 Ki = 1145 nM T83011 C1HM0I 17391146 IC50 = 1730 nM T83011 C56GJX 17391147 IC50 = 140.52 nM T83011 C61KJG 17391423 IC50 = 1920 nM T83011 CGIP10 17391461 IC50 = 1060 nM T83011 CK72SQ 17392369 IC50 = 271 nM T83011 C2LP8V 17462470 IC50 = 2023 nM T83011 CUTY36 17469896 IC50 = 616 nM T83011 CQ95CF 17471991 IC50 = 2790 nM T83011 CLR26X 17545843 IC50 = 490.84 nM T83011 CWI2E7 17738342 IC50 = 19070 nM T83011 C1QV5L 17738506 IC50 = 7090 nM T83011 CHZ0P1 17749832 IC50 = 6806 nM T83011 C0LAC8 17839878 IC50 = 8390 nM T83011 CO0BT3 18087653 IC50 = 8400 nM T83011 CC54WV 18093825 Ki = 294 nM T83011 CQ32FM 18151760 IC50 = 11600 nM T83011 CBD6Y7 18526002 IC50 = 510840 nM T83011 CRZI87 18943257 IC50 = 1140 nM T83011 C4SO6A 19132781 IC50 = 2650 nM T83011 CZTM17 19132783 IC50 = 351 nM T83011 C2Z6VI 19133248 IC50 = 14710 nM T83011 CI5LJ1 19133249 IC50 = 257.04 nM T83011 C34IVD 19133250 IC50 = 5477 nM T83011 CXR71E 19133252 IC50 = 2520 nM T83011 CMGL84 19133253 IC50 = 362 nM T83011 CBZ2J6 19133254 IC50 = 237 nM T83011 CX9AL2 19133255 IC50 = 2411 nM T83011 C26HDA 19133257 IC50 = 31197 nM T83011 C9ACO3 19133259 IC50 = 11530 nM T83011 CP98TF 19133260 IC50 = 43.65 nM T83011 C68VCD 19167136 IC50 = 937 nM T83011 C9V4ET 19204592 IC50 = 3750 nM T83011 C92UIL 19204597 IC50 = 9.47 nM T83011 CBLU27 19204599 IC50 = 61.2 nM T83011 CC85YA 19382380 IC50 = 20900 nM T83011 CJ1GF9 19556945 Ki = 310 nM T83011 C76DUN 19752124 IC50 = 17.38 nM T83011 C41BSF 20252235 IC50 = 10400 nM T83011 CR2V8K 20331466 IC50 = 6.2 nM T83011 C3DLC8 20404853 IC50 = 7300 nM T83011 C8B9FO 20438759 IC50 = 1400 nM T83011 CEJ36U 20559176 IC50 = 17970 nM T83011 CK27BD 20740795 Ki = 40 nM T83011 C05XEP 21239588 IC50 = 56120 nM T83011 CJX4A2 21240024 IC50 = 2230 nM T83011 C4EDK3 21671938 IC50 > 50000 nM T83011 C5I7VP 21964486 IC50 = 27.3 nM T83011 C0UK7W 21964497 IC50 = 43.2 nM T83011 CQ81MU 21964538 IC50 = 183 nM T83011 CTM62N 21974910 Ki = 9600 nM T83011 C5VJ4X 21982105 IC50 = 55.63 nM T83011 C2K4WS 22011729 IC50 = 1.9 nM T83011 C5YSK9 22055258 IC50 = 2483 nM T83011 CTC8J6 22215549 IC50 > 50000 nM T83011 CCJ4B7 22327634 IC50 = 140 nM T83011 CZ7L3Q 22421276 IC50 = 62 nM T83011 CJNT68 22569785 IC50 = 271900 nM T83011 CI30XB 22576850 IC50 = 5160 nM T83011 C2F6MQ 22601752 IC50 = 760 nM T83011 C81HXB 23372523 IC50 = 3225 nM T83011 CYOH73 23454034 IC50 = 6200 nM T83011 CN7LP5 23661731 IC50 = 2860 nM T83011 C7PK3S 23857007 IC50 = 6100 nM T83011 C5NXV3 23857375 IC50 = 6900 nM T83011 C9Y2EC 23879759 IC50 = 4 nM T83011 CV9DR5 23913004 IC50 = 1960 nM T83011 C3MEW7 23994505 IC50 = 9210 nM T83011 C21XUN 23996002 IC50 = 2.1 nM T83011 C2VR3X 24001527 IC50 = 8300 nM T83011 CSJ2B6 24164753 IC50 = 144 nM T83011 C9R1PK 24180717 IC50 = 72000 nM T83011 C5PG7Y 24230625 IC50 = 275 nM T83011 C58IBL 24395421 IC50 = 289 nM T83011 CR1L8S 24397125 IC50 = 407 nM T83011 CX98YL 24506542 IC50 = 449 nM T83011 CQZ20A 24506553 IC50 = 200 nM T83011 CT74EP 24689611 IC50 = 96.3 nM T83011 CTGB25 24695698 IC50 = 104 nM T83011 CL36IV 24709484 IC50 = 214 nM T83011 CDJ2C4 24709727 IC50 = 284 nM T83011 CM2J7N 24799761 IC50 = 1870 nM T83011 C36RNV 24860443 Ki = 1.17 nM T83011 C4CO3J 24860444 IC50 = 11.08 nM T83011 C9ZS8C 24860446 IC50 = 7.52 nM T83011 CNX32B 24860447 IC50 = 13.9 nM T83011 C6BUH8 24893999 IC50 = 1.18 nM T83011 C80WUR 24894016 IC50 = 160 nM T83011 CXRN67 25027416 IC50 = 64 nM T83011 C6ERN5 25027417 IC50 = 76 nM T83011 CCZ72B 25027418 IC50 = 2330 nM T83011 C9PY4E 25027421 IC50 = 2630.27 nM T83011 C9K0YJ 25034467 IC50 = 47.24 nM T83011 CH0M8Q 25034468 IC50 = 22.01 nM T83011 C97SXU 25034469 IC50 = 36.06 nM T83011 C5GAV4 25034470 IC50 = 30.08 nM T83011 CVNZ40 25034471 IC50 = 16.6 nM T83011 C0I8EP 25034472 IC50 = 9.8 nM T83011 CASW39 25034473 IC50 = 63.02 nM T83011 CN6DF9 25034474 IC50 = 32.48 nM T83011 C4MYE1 25139468 IC50 = 236 nM T83011 CANL42 25139470 IC50 = 260000 nM T83011 C7O1DP 25139471 IC50 = 44100 nM T83011 CA38ZR 25139472 IC50 = 10600 nM T83011 C5G4MN 25139474 IC50 = 73200 nM T83011 CI2GX7 25193423 IC50 = 162.18 nM T83011 C7VG9E 25193523 IC50 = 211 nM T83011 CD1YG4 25193524 IC50 = 13120 nM T83011 CD04UK 25193525 IC50 = 21900 nM T83011 C5B7XI 25193526 IC50 = 9550 nM T83011 CNW97L 25193527 IC50 = 5011.87 nM T83011 CJP69X 25193530 IC50 = 262 nM T83011 CS10DN 25193635 IC50 = 11956 nM T83011 C93CIO 25193636 IC50 = 2370 nM T83011 C54USH 25193637 IC50 = 4510 nM T83011 CF69VX 25193638 IC50 = 3120 nM T83011 C63AJF 25193733 IC50 = 477 nM T83011 C3HY2K 25194917 IC50 = 32.33 nM T83011 CP4LK1 25221889 IC50 > 100000 nM T83011 CL23IW 25254728 IC50 > 20000 nM T83011 CRK3Y8 25769005 IC50 > 50000 nM T83011 C1CK8A 26216970 IC50 = 1108 nM T83011 C5GRW1 26564219 IC50 = 642 nM T83011 C0KCL1 28369336 IC50 = 34.2 nM T83011 C13FZP 28369337 IC50 = 193 nM T83011 CZU47E 28369338 IC50 = 893 nM T83011 CTO2F8 28554530 IC50 = 1980 nM T83011 CLZ8F5 28739530 IC50 = 41900 nM T83011 C9FCN4 28825654 IC50 = 21.2 nM T83011 C82UJE 29283303 IC50 = 350 nM T83011 CL89DY 35793912 IC50 = 6900 nM T83011 CR6A9X 38763705 IC50 = 90 nM T83011 CE0G5M 38770453 IC50 = 59 nM T83011 CU04HR 39082892 Ki = 59 nM T83011 CRH7M4 39247144 Ki = 28 nM T83011 CZF25S 40041829 IC50 = 1700 nM T83011 CFYI84 42601491 IC50 = 1640 nM T83011 CP9K8Z 42618000 IC50 = 1030 nM T83011 C2FN1S 42618001 IC50 = 1258925.41 nM T83011 CQK9E4 42618002 IC50 = 71 nM T83011 C0VQH4 42618005 IC50 = 1.4 nM T83011 C7VKO3 42618006 IC50 = 9230 nM T83011 CO7Q8C 42618007 IC50 = 64450 nM T83011 C7V8UM 42618009 IC50 = 9590 nM T83011 CG8AX1 42618010 IC50 = 3690 nM T83011 CCW65K 42618011 IC50 = 16540 nM T83011 C58OWA 42618012 IC50 = 63520 nM T83011 C45TRB 42618013 IC50 = 61490 nM T83011 CX09CQ 42618014 IC50 = 4390 nM T83011 CP2QK3 42618015 IC50 = 3360 nM T83011 C8T3MQ 42618016 IC50 = 990 nM T83011 C8BL6I 42618017 IC50 = 4520 nM T83011 C5VNE8 42618018 IC50 = 3450 nM T83011 C19ICQ 42618020 IC50 = 41640 nM T83011 CGE5Q6 42618021 IC50 = 2870 nM T83011 CN38VU 42618022 IC50 = 21560 nM T83011 C3Q6VH 42618024 IC50 = 2370 nM T83011 C3N1XH 42618025 IC50 = 4980 nM T83011 C7HG2X 42623114 IC50 = 2210 nM T83011 CUEJ23 42623116 IC50 = 18990 nM T83011 CT9LN0 42623192 IC50 = 10960 nM T83011 C8EK3R 42623200 IC50 = 1610 nM T83011 CJ4MD2 42623269 IC50 = 1120 nM T83011 CCAW14 42623272 IC50 = 6430 nM T83011 CQ40TO 42623611 IC50 = 70 nM T83011 C5N7SE 42624010 IC50 = 180 nM T83011 CT1ND7 42624011 IC50 = 130 nM T83011 CN96DS 42624091 IC50 = 310 nM T83011 CXU9W0 42624092 IC50 > 30000 nM T83011 C6WVE8 42624093 IC50 = 90 nM T83011 C1QAC5 42624094 IC50 = 10 nM T83011 C7SE6I 42624095 IC50 = 6400 nM T83011 CZ0T8M 42624097 IC50 = 30 nM T83011 CPB14W 42624186 IC50 = 620 nM T83011 CEF0Y7 42624190 IC50 = 450 nM T83011 CCGY96 42624286 IC50 = 160 nM T83011 CJR34E 43090939 IC50 = 637 nM T83011 CDV3A8 43835789 IC50 = 127.4 nM T83011 CD0N4Z 44178231 IC50 = 145 nM T83011 COI86D 44221695 IC50 = 72.2 nM T83011 C7PI1S 44224195 IC50 = 8.98 nM T83011 C7EW5Z 44286698 Ki = 2300000 nM T83011 C6XMK4 44296124 IC50 = 19000 nM T83011 CSKW13 44296277 IC50 = 12 nM T83011 CWI9Y5 44296278 IC50 = 20 nM T83011 CIV34P 44345340 IC50 = 1513.56 nM T83011 CX05GA 44345341 IC50 = 1698.24 nM T83011 C2CBD8 44362199 IC50 = 57.54 nM T83011 C7PO9K 44362219 IC50 = 64.57 nM T83011 C6I1KB 44362434 IC50 = 1.096 nM T83011 CTL1W4 44362487 IC50 = 1.95 nM T83011 CDJC64 44362531 IC50 = 38 nM T83011 C52LPH 44371758 IC50 > 1000000 nM T83011 C9LZ3A 44371762 IC50 > 1000000 nM T83011 CS6Y9L 44371770 IC50 > 1000000 nM T83011 C9S8PR 44371772 IC50 > 1000000 nM T83011 CW2O7E 44371784 IC50 > 1000000 nM T83011 COX76Y 44371839 IC50 > 1000000 nM T83011 CX1TC7 44371843 IC50 = 317000 nM T83011 C2TI1K 44371844 IC50 > 1000000 nM T83011 CNZ59L 44371845 IC50 > 1000000 nM T83011 C5S4VL 44371849 IC50 = 77600 nM T83011 CB6L5H 44371855 IC50 > 1000000 nM T83011 C7X0ZU 44371902 IC50 = 51000 nM T83011 C81QMK 44371903 IC50 = 175000 nM T83011 CYPL76 44371904 IC50 > 1000000 nM T83011 CFQ15B 44371906 IC50 > 1000000 nM T83011 CY5E0V 44371918 IC50 = 395000 nM T83011 CI25TC 44371926 IC50 > 1000000 nM T83011 CPZ38Y 44372077 IC50 > 1000000 nM T83011 C1K8SH 44372226 Ki = 291000 nM T83011 C5WP7R 44376227 IC50 = 18 nM T83011 CLU6X0 44376584 IC50 = 20 nM T83011 CBN0X5 44376915 IC50 = 9 nM T83011 CYZ96F 44398186 Ki = 42000 nM T83011 C29VGR 44398252 Ki = 500000 nM T83011 CNW1H0 44398258 Ki > 100000 nM T83011 C3O7UN 44398289 Ki > 100000 nM T83011 CTIH68 44398308 Ki > 100000 nM T83011 C37ZKJ 44398338 Ki = 875000 nM T83011 CRPN02 44398339 Ki = 600000 nM T83011 CL23OZ 44398390 Ki = 10000 nM T83011 CI1LO2 44398465 Ki > 100000 nM T83011 C9T7SB 44398547 Ki > 100000 nM T83011 CZ0Q2P 44404688 Ki = 100000 nM T83011 CYTW05 44418972 IC50 = 710 nM T83011 C67ZNA 44437460 IC50 = 344 nM T83011 C6PK0B 44442374 IC50 = 134 nM T83011 CQ16OE 44442375 IC50 = 95 nM T83011 CG4SR1 44442378 IC50 = 142 nM T83011 CSX23C 44442379 IC50 = 2370 nM T83011 CI1XD0 44448000 IC50 = 32000 nM T83011 CMI7C5 44448037 IC50 = 4240 nM T83011 CIL0J4 44562978 IC50 = 856000 nM T83011 CEGS18 44563022 IC50 = 12980 nM T83011 C59WQS 44565882 IC50 = 4010 nM T83011 CV21MX 44577626 IC50 = 5400 nM T83011 CB1V4I 44577717 IC50 = 7100 nM T83011 CL2TP4 44577718 IC50 = 5100 nM T83011 CT9GO4 44577748 IC50 = 230000 nM T83011 CV45BR 44577749 IC50 = 470000 nM T83011 CU4T3C 44579922 Ki = 83 nM T83011 CX0OW8 44579936 Ki = 36000 nM T83011 C47HXL 44580006 Ki = 36 nM T83011 CQ16OW 44582853 IC50 = 2230 nM T83011 C47EYV 44587515 IC50 = 203.83 nM T83011 CT9VY0 44587516 IC50 = 26810 nM T83011 C2WV6H 44587534 IC50 = 14.2 nM T83011 CM2AF0 44587535 IC50 = 142.64 nM T83011 CWR84V 44587536 IC50 = 26.23 nM T83011 CU6S7O 44607264 IC50 = 500000 nM T83011 COW48M 44665667 IC50 = 1790 nM T83011 C7ZJH9 44886703 IC50 = 2320 nM T83011 CZ0QJ7 45113789 IC50 = 7180 nM T83011 CR53SL 45113790 IC50 = 18260 nM T83011 CLO07X 45113791 IC50 = 23210 nM T83011 C2QS6J 45113792 IC50 = 16330 nM T83011 C0P8RX 45113793 IC50 = 29380 nM T83011 C5YKT8 45113794 IC50 = 54510 nM T83011 CB8ZS5 45113924 IC50 = 2750 nM T83011 CM19RV 45113925 IC50 = 33260 nM T83011 CAPB61 45268543 IC50 = 40000 nM T83011 CH4NL1 45376336 IC50 = 1330 nM T83011 CNL38T 45490311 IC50 = 1790 nM T83011 CR8T0C 45490312 IC50 > 100000 nM T83011 CNY8M1 45906922 Ki = 550 nM T83011 C4EN8L 46222450 IC50 > 150000 nM T83011 CI0U9V 46223339 IC50 = 1000 nM T83011 CBV4W8 46232009 IC50 = 3340 nM T83011 C1JEG9 46236753 IC50 = 9000 nM T83011 CZO29G 46352302 IC50 = 121.62 nM T83011 C09EFO 46467419 Ki = 8010 nM T83011 C9HKJ2 46779222 IC50 = 10 nM T83011 C1FN3T 46830229 Ki > 133000 nM T83011 C72IST 46830246 IC50 = 8980 nM T83011 C48UBP 46847345 IC50 = 0.74 nM T83011 CV9DG4 46865967 IC50 = 160.64 nM T83011 CS6W7J 46889939 IC50 = 10000 nM T83011 CF7T8R 46895501 IC50 = 0.134 nM T83011 C2ZTX9 46933991 IC50 = 7120 nM T83011 CI7TL1 46944671 Ki = 39860 nM T83011 C8WH1R 46944673 Ki = 3830 nM T83011 C2FT5S 46944674 Ki = 430 nM T83011 CO7A5T 46944675 Ki = 520 nM T83011 C63XJZ 46944676 Ki = 190 nM T83011 C3I8WN 46945877 IC50 = 980000 nM T83011 CG58TS 46945878 IC50 = 72000 nM T83011 CT3IQ0 46945880 IC50 = 95000 nM T83011 CE95LB 46945881 IC50 = 86000 nM T83011 CKD6L8 46946079 IC50 = 240000 nM T83011 CN7DA6 46946080 IC50 = 380000 nM T83011 CV08XW 46946081 IC50 = 85000 nM T83011 CEFW62 46946082 IC50 = 7300000 nM T83011 C0VLP8 46946083 IC50 = 230000 nM T83011 CUFK84 46946084 IC50 = 940000 nM T83011 CA80DH 46946273 IC50 = 73000 nM T83011 CJI51A 46946280 IC50 = 15470 nM T83011 C6K8VD 46946463 IC50 = 18140 nM T83011 CS6PG9 46946464 IC50 = 50950 nM T83011 CN6YU8 46946465 IC50 = 53380 nM T83011 CMOF29 46946467 IC50 = 71300 nM T83011 CT1DY2 46946469 IC50 = 13700 nM T83011 C3JFT7 46946470 IC50 = 16770 nM T83011 C1KZW6 46946666 IC50 = 49440 nM T83011 C0RN8K 46946667 IC50 = 84640 nM T83011 CW61BI 46946671 IC50 = 34810 nM T83011 CU8G7X 46947641 Ki = 4230 nM T83011 C3OK9X 46947642 Ki = 75720 nM T83011 C1CAN0 46949549 IC50 = 821 nM T83011 C5E6XN 47002592 IC50 > 10000 nM T83011 C9HW8B 47003377 IC50 = 926 nM T83011 CC81EY 47398190 IC50 = 86 nM T83011 CJ29HG 47420565 IC50 = 620 nM T83011 CT3I6B 48036542 IC50 = 69.51 nM T83011 C3DK8H 49098177 IC50 = 1170 nM T83011 CA6SL4 49863576 IC50 = 231.02 nM T83011 C87CZL 49863577 IC50 = 26.64 nM T83011 CG5L1Q 49863578 IC50 = 1060 nM T83011 CU54BX 49863607 IC50 = 31.87 nM T83011 CJW3D5 49863635 IC50 = 12.22 nM T83011 C9TL2A 49863636 IC50 = 72.7 nM T83011 CF9TR0 49863637 IC50 = 35.49 nM T83011 COR75I 49863638 IC50 = 29.54 nM T83011 CVX08W 49863730 IC50 = 6970 nM T83011 C52UHN 49864177 IC50 > 1000000 nM T83011 CPO5C2 49864508 IC50 = 4890 nM T83011 C35XSM 49868483 Ki = 17000 nM T83011 CU5XE6 50745004 IC50 > 100000 nM T83011 CO35KG 50876171 IC50 = 3190 nM T83011 C2X9QA 50876174 IC50 = 3.802 nM T83011 CS96UB 50994176 Ki = 0.28 nM T83011 CBA14N 51003565 IC50 = 7.943 nM T83011 C8BL3V 51003566 IC50 = 11.48 nM T83011 C35DLK 51049245 IC50 = 56800 nM T83011 CM73OT 51223711 IC50 = 9800 nM T83011 C4Q6RF 52174704 IC50 = 164 nM T83011 C38DBE 52446186 IC50 = 2118 nM T83011 C2DBZ5 52541425 IC50 = 288 nM T83011 CU5E0F 52643177 IC50 = 550 nM T83011 CO96MS 52913781 IC50 = 930 nM T83011 C9KRJ8 52913782 IC50 = 37690 nM T83011 CH5X8F 52915137 IC50 = 1920 nM T83011 CFYQ13 52915138 IC50 = 45.95 nM T83011 C4X7AT 52915139 IC50 = 633.55 nM T83011 CIS6D4 52915140 IC50 = 233.73 nM T83011 C0FTO3 52936300 IC50 = 483.88 nM T83011 C8QCO0 52937825 IC50 = 331.11 nM T83011 CWVC67 52937826 IC50 = 870963.59 nM T83011 C8TRH1 52940770 IC50 = 36 nM T83011 CVY9C7 52940812 IC50 = 120 nM T83011 C7NUM5 52941235 IC50 = 940 nM T83011 C81FZE 52941812 IC50 = 2230 nM T83011 C0HVE2 52941960 IC50 = 86 nM T83011 CO42IY 52942005 IC50 = 200 nM T83011 CO6R7T 52942020 IC50 = 410 nM T83011 C14CJD 52942390 IC50 = 40.74 nM T83011 C09WXG 52942474 IC50 = 912.01 nM T83011 C0J2FL 52943064 IC50 = 115920 nM T83011 C0CB3Z 52943176 IC50 = 30 nM T83011 C4O7NQ 52943178 IC50 = 210 nM T83011 CW86YM 52943217 IC50 = 3680 nM T83011 CX0Y2K 52943218 IC50 = 56 nM T83011 C0HVJ6 52943230 IC50 = 26 nM T83011 CP5NZ8 52943354 IC50 = 652 nM T83011 CL94WN 52943606 IC50 = 3 nM T83011 C7R0ZB 52944251 IC50 = 62070 nM T83011 CJKO37 52944406 IC50 = 9 nM T83011 C49EYX 52944409 IC50 = 150 nM T83011 C98VBM 52945642 IC50 = 20 nM T83011 CD40XF 52945645 IC50 = 47 nM T83011 CI9Y4H 52945649 IC50 = 260 nM T83011 C6JKN7 52945917 IC50 = 91.2 nM T83011 CBD1G2 52946045 IC50 = 61.66 nM T83011 CD85UQ 52946066 IC50 = 3.548 nM T83011 CJX6E9 52946067 IC50 = 16 nM T83011 CP51KJ 52946520 IC50 = 17 nM T83011 CJ7SQ1 52946862 IC50 = 18 nM T83011 C5NQ0L 52946864 IC50 = 230 nM T83011 C2EQ0Z 52947352 IC50 = 45.71 nM T83011 CO0D3Z 52947695 IC50 = 85.11 nM T83011 CUP46C 52948039 IC50 = 410 nM T83011 CG9X5N 52948086 IC50 = 32 nM T83011 CZIW51 52948923 IC50 = 810 nM T83011 CM2H4L 52949147 IC50 = 56880 nM T83011 C12DYG 52949244 IC50 = 14 nM T83011 CKE8D5 52949315 IC50 = 13126 nM T83011 CM9B7Z 52949317 IC50 = 26810 nM T83011 C6S4IX 52949319 IC50 = 32 nM T83011 C89GLO 52949320 IC50 = 9650 nM T83011 CS32GV 52949324 IC50 = 420 nM T83011 CS9NO2 52949516 IC50 = 52.48 nM T83011 CJC20G 52949550 IC50 = 9446 nM T83011 CK15PD 52950170 IC50 = 63 nM T83011 CGQ76K 53009757 IC50 = 571 nM T83011 CJQ24Z 53019680 IC50 = 115.31 nM T83011 CDHY42 53248703 IC50 = 30910 nM T83011 CVZ2D4 53248704 IC50 = 16870 nM T83011 C6Z0BI 53315284 IC50 = 60 nM T83011 CP39IR 53317196 Ki = 28 nM T83011 CNFA87 53318409 IC50 = 52.65 nM T83011 CBN96D 53319414 IC50 = 120 nM T83011 C9UD2P 53319928 Ki = 603 nM T83011 CH38CS 53320714 IC50 = 450 nM T83011 CKZ0C3 53322381 IC50 = 12.34 nM T83011 CW81FC 53322432 Ki = 4280 nM T83011 C12ZPO 53323736 IC50 = 35.26 nM T83011 C4A3YO 53323737 IC50 = 51.37 nM T83011 CI6TF9 53358323 IC50 = 1.35 nM T83011 C76GDP 53358665 Ki = 4790 nM T83011 CIVP93 53361170 Ki = 280 nM T83011 C5BM2I 53361171 Ki = 280 nM T83011 CQ2Z4F 53361172 Ki = 88 nM T83011 CUI4C7 53361173 Ki = 45 nM T83011 C19YQZ 53361174 Ki = 48 nM T83011 C6Z0DN 53375709 Ki = 2190 nM T83011 C7PNY9 53375710 Ki = 11650 nM T83011 CHNB31 53375711 Ki = 2760 nM T83011 C89TBV 53375712 Ki = 130 nM T83011 C5PN6W 53375893 IC50 = 3770 nM T83011 CJ56PN 53380594 IC50 = 110 nM T83011 C1H4LY 53387407 IC50 = 1080 nM T83011 C7TM8P 53387408 IC50 = 11780 nM T83011 CKCG05 53392601 IC50 = 340 nM T83011 C2SL6G 53465287 IC50 = 100.64 nM T83011 C4CS0K 53465288 IC50 = 8460 nM T83011 CVS5J9 53465289 IC50 = 82.54 nM T83011 CKH85U 53484089 Ki = 3 nM T83011 CY3F4K 53484090 Ki = 29 nM T83011 C5VKC4 53484091 Ki = 10 nM T83011 CPKR28 53484109 Ki = 24 nM T83011 C0VD5I 54327402 IC50 = 812500 nM T83011 C5I7JA 54526203 IC50 = 3530 nM T83011 CB16CK 54578559 IC50 = 46820 nM T83011 CA8WX6 54579011 IC50 = 220.61 nM T83011 CWL96S 54579012 IC50 = 9530 nM T83011 CYH7N1 54579013 IC50 = 19360 nM T83011 CGC15Z 54580315 IC50 = 262.95 nM T83011 CTM81X 54580620 IC50 = 83.48 nM T83011 CD01OR 54690405 IC50 = 69590 nM T83011 C6D9IE 54753443 IC50 = 32 nM T83011 CR61HF 54753444 IC50 = 26 nM T83011 C69HSF 54770057 Ki = 32 nM T83011 CAG3F4 55285162 IC50 = 10 nM T83011 CLRG73 55327852 IC50 = 7070 nM T83011 CIGK63 55471034 IC50 = 531 nM T83011 CYC5V0 55471035 IC50 = 484 nM T83011 CG70OK 56594086 IC50 = 17.05 nM T83011 C9N7HQ 56594087 IC50 = 1.52 nM T83011 C5R1CX 56594088 IC50 = 67.1 nM T83011 CO7VE3 56594089 IC50 = 5520 nM T83011 C5DEQ8 56594090 IC50 = 14470 nM T83011 C7ZLC4 56594232 IC50 = 15.01 nM T83011 C8JOY4 56594233 IC50 = 3.25 nM T83011 C9OI3Q 56594234 IC50 = 54030 nM T83011 CI8F9G 56594236 IC50 = 650.03 nM T83011 C54NUW 56594237 IC50 = 120.02 nM T83011 CKJ8D0 56594370 IC50 = 180.04 nM T83011 CBX47T 56603017 IC50 = 5 nM T83011 CM4UH3 56640830 IC50 = 8620 nM T83011 CU1T2L 56640833 IC50 = 1190 nM T83011 CJ8O3M 56640990 IC50 = 6650 nM T83011 C93UAM 56640991 IC50 = 2200 nM T83011 C5X8JV 56640992 IC50 = 2730 nM T83011 CD0ST5 56640993 IC50 = 48100 nM T83011 C0JXD8 56640994 IC50 = 23500 nM T83011 CDU32V 56640995 IC50 = 30900 nM T83011 CMTZ92 56640996 IC50 = 1010 nM T83011 CMVU62 56642649 IC50 = 140 nM T83011 CQL3T5 56642783 IC50 = 21.47 nM T83011 CDR4G1 56642784 IC50 = 1800 nM T83011 C25NAV 56642786 IC50 = 410 nM T83011 CC9L2R 56649563 Ki = 110 nM T83011 CK0SB8 56659353 Ki = 7 nM T83011 CE2BN7 56659354 Ki = 20 nM T83011 C2N1XU 56659718 Ki = 22000 nM T83011 CN7W5K 56659719 Ki = 3200 nM T83011 CP36XA 56662172 IC50 = 16060 nM T83011 C5WM4L 56663182 Ki = 400900 nM T83011 CVP6U5 56665630 IC50 = 31650 nM T83011 CSW8C3 56666850 IC50 = 17510 nM T83011 CFL96D 56668520 IC50 = 56000 nM T83011 C9EX4Z 56670040 Ki = 300010 nM T83011 C24DGB 56670041 Ki = 1660 nM T83011 CTM1D9 56670052 IC50 = 73920 nM T83011 CA50XS 56670279 IC50 = 27110 nM T83011 CD84RE 56670280 IC50 = 14810 nM T83011 C6CN3P 56673197 Ki = 20 nM T83011 CZQ8I0 56673343 Ki = 355000 nM T83011 CR4BD5 56673554 Ki = 250000 nM T83011 CU7FR3 56673555 Ki = 60000 nM T83011 CVRQ94 56673556 Ki = 4800 nM T83011 CUD04Q 56676876 Ki = 979000 nM T83011 CBX28Q 56676877 Ki = 255600 nM T83011 C3UEL1 56680195 Ki = 2130000 nM T83011 C2LV9D 56683530 Ki = 309220 nM T83011 CC8A4B 56683531 Ki = 4000 nM T83011 CH1LS7 56683532 Ki = 4110 nM T83011 CEML01 56683533 Ki = 4220 nM T83011 COLW37 56709688 IC50 = 42500 nM T83011 CXI01A 56807126 IC50 = 2100 nM T83011 C4YFN8 56834983 IC50 = 2790 nM T83011 CPZ6T7 56933768 Ki = 480 nM T83011 C0VI8M 56950927 IC50 = 167 nM T83011 C81FBW 56966263 IC50 = 768 nM T83011 CXD3C0 57303200 IC50 = 17800 nM T83011 CRF07B 57325839 IC50 = 62 nM T83011 C4RG0D 57328315 IC50 = 27 nM T83011 C8TN7H 57335751 IC50 = 3830 nM T83011 CN28HO 57340730 IC50 = 642 nM T83011 C7L2FP 57340731 IC50 = 4.8 nM T83011 CE6LJ1 57379747 IC50 = 21 nM T83011 CJ12FR 57379748 IC50 = 57 nM T83011 CVW96L 57379749 IC50 = 3.6 nM T83011 C60GZY 57379750 IC50 = 2 nM T83011 CCED62 57379751 IC50 = 2 nM T83011 C28HTP 57379977 IC50 = 3.3 nM T83011 CM72YD 57379978 IC50 = 13 nM T83011 CAE03J 57379979 IC50 = 8.4 nM T83011 CG43VX 57379980 IC50 = 19 nM T83011 C16SCD 57379981 IC50 = 6 nM T83011 CN0L3H 57379982 IC50 = 76 nM T83011 COX83F 57379983 IC50 = 22 nM T83011 C94HLT 57379984 IC50 = 2 nM T83011 CCD0W7 57380218 IC50 = 27 nM T83011 CP3R2T 57387314 IC50 > 10000 nM T83011 CQW5T3 57387397 IC50 = 91.8 nM T83011 COZ7L2 57388814 IC50 = 77.9 nM T83011 C3MOX5 57388817 IC50 = 71.8 nM T83011 CR87KW 57388819 IC50 = 927 nM T83011 C08OQJ 57388899 IC50 = 4.5 nM T83011 CUOT05 57388979 IC50 = 65 nM T83011 CY5S1I 57389059 IC50 = 34.4 nM T83011 CQRM60 57390487 IC50 = 19400 nM T83011 CGSX75 57392339 IC50 = 223 nM T83011 C1PJO0 57392340 IC50 = 13100 nM T83011 CZ53IA 57392341 IC50 = 3600 nM T83011 C3XO9E 57392561 IC50 = 1580 nM T83011 C0RUX5 57392562 IC50 = 1540 nM T83011 CG5AM8 57392798 IC50 > 2000 nM T83011 CRAF46 57392799 IC50 = 170.5 nM T83011 C2COB9 57394022 IC50 = 24400 nM T83011 C54XIL 57394023 IC50 = 2970 nM T83011 C0Z7SL 57396037 IC50 = 2530 nM T83011 C3CWN6 57397563 IC50 = 9600 nM T83011 CZ90QM 57397635 IC50 = 332 nM T83011 CG5N1V 57397741 Ki > 40000 nM T83011 C6A1YR 57397784 IC50 = 96100 nM T83011 CKST71 57397880 IC50 = 42680 nM T83011 CIV67J 57398073 IC50 > 2000 nM T83011 CTV5M3 57399451 IC50 = 1362900 nM T83011 CC5JQ1 57399500 IC50 = 3650 nM T83011 CL8FQ1 57399501 IC50 = 11700 nM T83011 CIY0U2 57399502 IC50 = 150 nM T83011 CH47EP 57399503 IC50 = 4300 nM T83011 CY1S3R 57399530 IC50 = 9260 nM T83011 C9PE1R 57401006 IC50 = 16800 nM T83011 CW9R4F 57401210 IC50 = 5265900 nM T83011 CQ1D3R 57401211 IC50 = 67200 nM T83011 C5ZBW3 57401260 IC50 = 10800 nM T83011 CR12SB 57401261 IC50 = 2250 nM T83011 CIQ3W0 57401289 IC50 = 32040 nM T83011 CJ3RM8 57402930 Ki = 7400 nM T83011 C3NP9V 57402959 IC50 = 1245100 nM T83011 C5VT3D 57789264 IC50 = 27 nM T83011 C2R5US 58495647 IC50 = 4770 nM T83011 C7FBJ5 59165653 IC50 = 15600 nM T83011 C1HS5X 59588962 IC50 = 30 nM T83011 C3NFG6 59588969 IC50 = 2980 nM T83011 C1DER5 59601689 IC50 = 861 nM T83011 CV3JF1 59976344 IC50 = 20200 nM T83011 C68XHY 60161811 IC50 > 10000 nM T83011 CD6B5P 60203904 IC50 = 1800 nM T83011 C2WQN8 60264513 IC50 = 96.51 nM T83011 COHF58 60264536 IC50 = 56.89 nM T83011 C3JYI8 60351355 IC50 = 109 nM T83011 CJYV91 60373147 IC50 = 248 nM T83011 CDF54K 60627106 IC50 = 8630 nM T83011 C2NRD5 60644162 IC50 = 19300 nM T83011 CL9DK6 60670209 IC50 = 300 nM T83011 CTH3G9 60714993 IC50 = 335 nM T83011 C3XC5K 60715051 IC50 = 234 nM T83011 CL9QK4 60715052 IC50 = 1300 nM T83011 C0ID4P 60715244 IC50 = 1280 nM T83011 C3Z4GX 60772162 IC50 = 20510 nM T83011 CCJ0Q9 61242666 IC50 = 316 nM T83011 C41OAY 61832262 IC50 = 17 nM T83011 CF87MH 61832641 IC50 = 11 nM T83011 C0L8SP 61832822 IC50 = 8 nM T83011 CMU52G 61833183 IC50 = 9 nM T83011 CS04ZK 61833537 IC50 = 32 nM T83011 CN54TI 61833721 IC50 = 11 nM T83011 C7BG9L 61833723 IC50 = 15 nM T83011 CDK32Q 61834439 IC50 = 9 nM T83011 CA7P8O 61834440 IC50 = 78 nM T83011 C0E8MG 63095539 IC50 = 2130 nM T83011 C60JPX 63718419 IC50 = 0.227 nM T83011 CL7R0T 63937924 IC50 < 10000 nM T83011 C17WZV 64789040 IC50 = 6220 nM T83011 C4RV3T 65477805 IC50 = 4.5 nM T83011 C1A3FG 66523802 IC50 = 625 nM T83011 CQTC83 66571530 IC50 = 79000 nM T83011 CCO53I 66571532 IC50 = 25000 nM T83011 CS7ZX1 66571590 IC50 = 25000 nM T83011 CO84GD 66712998 IC50 = 179 nM T83011 C1GXR4 69889948 IC50 = 3 nM T83011 C3PDQ5 70682249 IC50 = 576 nM T83011 CYG64Z 70682250 IC50 = 5.7 nM T83011 CZ71QR 70682919 IC50 = 190 nM T83011 CFYC13 70684340 IC50 = 77.4 nM T83011 CI5ZC4 70684852 IC50 = 1610 nM T83011 CY39PE 70684853 IC50 = 189 nM T83011 CW3TY2 70684854 IC50 = 18400 nM T83011 C7IG3N 70684855 IC50 = 124000 nM T83011 CAV03I 70684998 IC50 = 490 nM T83011 CYS03B 70686497 IC50 = 8030 nM T83011 CYM2D6 70686498 IC50 = 4340 nM T83011 CMW14V 70687001 IC50 = 825 nM T83011 CJNL16 70688596 IC50 = 172 nM T83011 CJ32UT 70689077 IC50 = 148 nM T83011 CYX4M9 70689078 IC50 = 641 nM T83011 C4G5FW 70689079 IC50 = 1230 nM T83011 CY05LV 70689080 IC50 = 108000 nM T83011 CT9FI6 70689081 IC50 = 5670 nM T83011 CI1Q2S 70689082 IC50 = 7790 nM T83011 C12QAY 70690656 IC50 = 2.8 nM T83011 C6NWQ7 70690657 IC50 = 5960 nM T83011 CCK52V 70691189 IC50 = 4050 nM T83011 CP3V7G 70691190 IC50 = 64100 nM T83011 C0M7EU 70692804 IC50 = 3.7 nM T83011 CAT52I 70692805 IC50 = 4 nM T83011 CIN7O4 70692806 IC50 = 4 nM T83011 C0RM9W 70693292 IC50 = 5780 nM T83011 CD5T8W 70693293 IC50 = 250 nM T83011 C9I3PY 70693294 IC50 = 6120 nM T83011 CQ9NO2 70694840 IC50 = 44800 nM T83011 CE36KZ 70695386 IC50 = 334 nM T83011 C7VGX8 70695387 IC50 = 4900 nM T83011 CQ4U0F 70695388 IC50 = 22300 nM T83011 CJBL13 70695389 IC50 = 17900 nM T83011 CB7R4L 70695390 IC50 = 8420 nM T83011 C3KFZ2 70695391 IC50 = 6910 nM T83011 CT8E7W 70696891 IC50 = 2690 nM T83011 CNR15V 70697409 IC50 = 23400 nM T83011 CYAS63 70697549 IC50 = 1240 nM T83011 CTFG16 70702063 IC50 = 17 nM T83011 CI69QM 70702068 IC50 = 25 nM T83011 CXLT46 70702073 IC50 = 27.82 nM T83011 C18MPL 70723639 IC50 > 200000 nM T83011 C7L6PQ 70804892 IC50 = 114 nM T83011 CR6D8Y 71256270 IC50 = 334.5 nM T83011 C3O2BL 71256276 IC50 = 267.1 nM T83011 CN5T6M 71256288 IC50 = 271.8 nM T83011 CU8R2W 71256323 IC50 = 356 nM T83011 CZB3U7 71256332 IC50 = 270.3 nM T83011 CTE2I3 71256340 IC50 = 1372.8 nM T83011 CON49H 71261649 IC50 > 20000 nM T83011 C7POG5 71263675 IC50 = 889.5 nM T83011 CR3BH2 71263683 IC50 = 2539.2 nM T83011 C2DI4G 71351539 IC50 > 50000 nM T83011 C2Q0VE 71419878 IC50 = 42.75 nM T83011 C42BYX 71449560 IC50 = 457 nM T83011 CQ3OZ8 71450450 IC50 = 14 nM T83011 CZ5H9R 71450578 IC50 = 17 nM T83011 CCW1Z5 71450579 IC50 = 227 nM T83011 C3FC2B 71450580 IC50 = 19 nM T83011 C2G1FO 71451363 IC50 = 6.8 nM T83011 COP81R 71451364 IC50 = 364 nM T83011 CWHM59 71452280 IC50 = 34 nM T83011 CLB25C 71452281 IC50 = 124 nM T83011 C6I2MP 71452416 IC50 = 72 nM T83011 C7F4XP 71452417 IC50 = 43 nM T83011 CLE84D 71452418 IC50 = 131000 nM T83011 C3ZD2F 71453027 IC50 = 1420 nM T83011 CK3G4B 71453169 IC50 = 7.4 nM T83011 C1T8YS 71454081 IC50 = 223 nM T83011 C1U2GV 71454184 IC50 = 51 nM T83011 C0CJV9 71454185 IC50 = 781 nM T83011 CBQ74P 71455816 IC50 = 1810 nM T83011 CEI09U 71455925 IC50 = 19 nM T83011 CJO48H 71455926 IC50 = 23 nM T83011 CJ4B2W 71456691 IC50 = 4.5 nM T83011 CJTE73 71456692 IC50 = 30 nM T83011 CQ6UP9 71457124 IC50 = 18550 nM T83011 CS5X1P 71457606 IC50 = 449 nM T83011 C87RFW 71457723 IC50 = 40 nM T83011 CRL5P4 71457724 IC50 = 125 nM T83011 CUIF34 71457725 IC50 = 61 nM T83011 C9UHF3 71458533 IC50 = 20 nM T83011 CBX0C4 71459629 IC50 = 71 nM T83011 CL0HS2 71459630 IC50 = 3500 nM T83011 C7I2JG 71459631 IC50 = 62 nM T83011 C8UJ0T 71460379 IC50 = 5.6 nM T83011 C4N8JG 71461236 IC50 = 25 nM T83011 C1L7MK 71461237 IC50 = 67 nM T83011 C7HA0O 71461238 IC50 = 79 nM T83011 CRPA65 71461239 IC50 = 887 nM T83011 C1PG9R 71461375 IC50 = 471 nM T83011 CL1FP5 71461376 Ki = 9.8 nM T83011 C85UCB 71462073 IC50 = 15 nM T83011 C9A6PQ 71462516 IC50 = 28700 nM T83011 C4PIQ9 71462518 IC50 = 40500 nM T83011 C6G4XF 71462972 IC50 = 242 nM T83011 CG01AM 71508602 IC50 = 664 nM T83011 CI1C7E 71508637 IC50 = 208.5 nM T83011 C36MKD 71508638 IC50 = 131.5 nM T83011 CJP68B 71543365 IC50 > 100000 nM T83011 CW2T6C 71559776 IC50 = 2.8 nM T83011 CVQ8S3 71559777 IC50 = 2.4 nM T83011 C9UM3S 71559778 IC50 = 6.4 nM T83011 CJ7O6M 71559779 Ki = 0.46 nM T83011 C2DM5F 71559780 IC50 = 1.8 nM T83011 CMZ38H 71559781 IC50 = 9 nM T83011 CCXO52 71559911 IC50 = 3.5 nM T83011 CSD8O4 71559912 IC50 = 47 nM T83011 C73IBL 71559913 IC50 = 48 nM T83011 CKH79U 71559914 IC50 = 68 nM T83011 C3RP6O 71559915 IC50 = 81 nM T83011 CEZ32S 71559916 IC50 = 18 nM T83011 CZS83E 71559917 IC50 = 11 nM T83011 C8NKJ7 71559918 IC50 = 12 nM T83011 CBHX24 71560037 IC50 = 7.4 nM T83011 CDO3U5 71560038 IC50 = 12 nM T83011 CZXY43 71561477 IC50 > 1000 nM T83011 C0FJ1X 71561478 IC50 = 173.2 nM T83011 CYZE35 71561479 IC50 = 67.8 nM T83011 C3QJ5M 71561480 IC50 > 1000 nM T83011 C65OJL 71561481 IC50 > 1000 nM T83011 CF4T7N 71561482 IC50 = 48.1 nM T83011 C13TRN 71561483 IC50 = 582.8 nM T83011 C43UWM 71561593 IC50 > 1000 nM T83011 C7CFR4 71561594 IC50 > 1000 nM T83011 C4YZ8I 71561595 IC50 > 10000 nM T83011 CYM5Q0 71561596 IC50 > 10000 nM T83011 C6XV7D 71562554 IC50 > 10000 nM T83011 CU8QC4 71562555 IC50 > 10000 nM T83011 C2GOS6 71562556 IC50 = 182.3 nM T83011 CH7A3C 71562557 IC50 > 1000 nM T83011 CI5JP8 71562669 IC50 > 10000 nM T83011 CN25AT 71562670 IC50 > 10000 nM T83011 CZG10K 71562924 IC50 = 7630 nM T83011 C1RQ0X 71562925 IC50 = 1390 nM T83011 CJ5M2B 71562926 IC50 = 5220 nM T83011 CH45VQ 71562928 IC50 = 1480 nM T83011 C3XTO4 71562929 IC50 = 370.2 nM T83011 C1SYX5 71563047 IC50 = 480 nM T83011 CX40FP 71563048 IC50 = 174.6 nM T83011 C2A9VU 71563049 IC50 = 200 nM T83011 CHVB51 71563050 IC50 = 431.5 nM T83011 C4N2XD 71563051 IC50 = 762.5 nM T83011 CL60DA 71563052 IC50 = 1368 nM T83011 C41JWM 71563053 IC50 = 266.7 nM T83011 CBD60O 71563170 IC50 = 132.9 nM T83011 C9PEA5 71563171 IC50 > 1000 nM T83011 CI74VT 71563173 IC50 > 10000 nM T83011 C5H3ZN 71563174 IC50 > 10000 nM T83011 C3UD6V 71563175 IC50 > 10000 nM T83011 C4DE7M 71563176 IC50 = 586.7 nM T83011 C64RSC 71563296 IC50 > 1000 nM T83011 C5DZM0 71563297 IC50 = 543.3 nM T83011 CSVQ36 71563298 IC50 > 10000 nM T83011 C2Z9RH 71563299 IC50 > 1000 nM T83011 C65EVL 71563300 IC50 > 10000 nM T83011 CQ2SL9 71563301 IC50 > 1000 nM T83011 C0PI4G 71563302 IC50 > 1000 nM T83011 C6OAN3 71568924 IC50 = 4.51 nM T83011 CU6NX9 71568925 IC50 = 11.35 nM T83011 CL19VB 71568926 IC50 = 725.92 nM T83011 CIQT69 71568927 IC50 = 14610 nM T83011 CY91WT 71568929 IC50 = 501.66 nM T83011 CSYG87 71569082 IC50 = 486.35 nM T83011 C26OKQ 71569083 IC50 = 1450 nM T83011 C6S5CK 71569084 IC50 = 969.44 nM T83011 C8DY4I 71589260 IC50 = 20080 nM T83011 CSM4W0 71616357 IC50 = 790700 nM T83011 CQ3I9J 71616361 IC50 > 1250000 nM T83011 CJTX03 71652416 IC50 = 11070 nM T83011 CK1FR2 71652417 IC50 = 6210 nM T83011 CK57NM 71652418 IC50 = 519 nM T83011 CJNR53 71652419 Ki = 0.129 nM T83011 C5HPG0 71652824 IC50 > 1250000 nM T83011 CA8BI9 71654261 IC50 = 18110 nM T83011 CA73CM 71654421 IC50 = 693 nM T83011 CM20YQ 71654422 IC50 = 4460 nM T83011 C4Y0SL 71654423 IC50 = 8550 nM T83011 C1TPO4 71654581 IC50 = 2400 nM T83011 C9HL6M 71654582 IC50 = 209 nM T83011 C6V1HF 71654583 IC50 = 167 nM T83011 C4D0WN 71654584 IC50 = 181 nM T83011 C79DOY 71654585 IC50 = 346 nM T83011 CK5Z8Q 71660500 IC50 = 45 nM T83011 C70SIG 71680729 IC50 = 1.63 nM T83011 C0YW1C 71680730 IC50 = 470 nM T83011 CG6EY1 71680731 IC50 = 93.3 nM T83011 CN0WU1 71680732 IC50 = 43.7 nM T83011 CK2Y6A 71680733 IC50 = 34.9 nM T83011 CH5KU9 71680734 IC50 = 389 nM T83011 C6OXR9 71680735 IC50 > 1000 nM T83011 CA50LT 71680889 IC50 = 3440 nM T83011 CCM92I 71680890 IC50 = 39.8 nM T83011 CS51FY 71680891 IC50 = 238 nM T83011 CX4BZ6 71680892 IC50 > 1000 nM T83011 CC7MA1 71680893 IC50 > 10000 nM T83011 C6HZ4O 71680894 IC50 > 10000 nM T83011 CN0EZ6 71680895 IC50 > 10000 nM T83011 C30NCG 71681049 IC50 > 10000 nM T83011 C2TR7P 71681050 IC50 = 53.1 nM T83011 CVY85K 71681051 IC50 = 94 nM T83011 C8TCR6 71681052 IC50 > 10000 nM T83011 C4KB8W 71681053 IC50 > 10000 nM T83011 CLBD58 71681054 IC50 = 76.4 nM T83011 C50TBU 71681055 IC50 = 206 nM T83011 C2Y3KO 71681203 IC50 = 69.7 nM T83011 CIM0S3 71681204 IC50 = 9.8 nM T83011 C21UWV 71683091 IC50 = 17.6 nM T83011 COWX82 71683092 IC50 = 95.3 nM T83011 C9CLQ3 71683093 IC50 > 10000 nM T83011 CV5O0H 71683094 IC50 = 11.2 nM T83011 CCJ17F 71683095 IC50 = 2.09 nM T83011 CY0OQ8 71716963 IC50 = 1460 nM T83011 C4EQA2 71717323 IC50 = 35481.34 nM T83011 CS51AY 71717592 IC50 = 160.32 nM T83011 CZY42C 71717593 IC50 = 153.14 nM T83011 C4BVA5 71717928 IC50 = 430.3 nM T83011 CP3GK8 71720004 IC50 = 1810 nM T83011 CG4PR6 71764406 IC50 = 12160 nM T83011 CI4Q6K 71764831 IC50 = 14090 nM T83011 CWXB75 71769421 IC50 = 665.1 nM T83011 C63VCE 71769543 IC50 = 171.4 nM T83011 C07KCU 71769544 IC50 = 357.9 nM T83011 CAV41T 71816334 IC50 = 6800 nM T83011 CLC90S 71818857 IC50 = 344 nM T83011 CP07TK 71818858 Ki = 144 nM T83011 CJ6ON9 71818859 IC50 = 206 nM T83011 C4LW8O 71818860 IC50 = 543 nM T83011 CB48KD 72164304 IC50 = 280 nM T83011 C5QO7E 72164305 IC50 = 60 nM T83011 CE6FJ2 72164306 IC50 = 140 nM T83011 CXQ0T2 72164307 IC50 = 110 nM T83011 CZ43TD 72164308 IC50 = 110 nM T83011 CN2XA3 72164426 IC50 = 3650 nM T83011 C4PB7G 72164427 IC50 = 840 nM T83011 CQJE58 72164428 IC50 = 3950 nM T83011 C1REN4 72191056 IC50 = 2330 nM T83011 CN56AJ 72191362 IC50 = 284 nM T83011 CHE87W 72191363 IC50 = 6.2 nM T83011 C3RYV1 72191364 Ki = 2.7 nM T83011 C81BYJ 72191365 IC50 = 191 nM T83011 CHL70P 72191366 IC50 = 130 nM T83011 C9M4CN 72196362 IC50 = 6630 nM T83011 CHT07I 72196364 IC50 = 5080 nM T83011 C27CBN 72206251 IC50 = 173 nM T83011 CS81LQ 72696144 IC50 > 10000 nM T83011 C3BEM8 72696145 IC50 = 62.9 nM T83011 C1E4ZD 72696146 IC50 = 193 nM T83011 CQ35NL 72696147 IC50 = 1350 nM T83011 CRN4B1 72696148 IC50 = 86.9 nM T83011 C0IF1J 72696149 IC50 = 10000 nM T83011 CL2H7Y 72696273 IC50 = 2200 nM T83011 C7MX9Y 72696274 IC50 = 10000 nM T83011 CBTE63 72696275 IC50 > 10000 nM T83011 CPI89R 72696276 IC50 = 3480 nM T83011 COX4B1 72696277 IC50 > 10000 nM T83011 CI9HP7 72696397 IC50 = 10000 nM T83011 C1RFY6 72696398 IC50 = 10000 nM T83011 CY56RG 72696399 IC50 > 10000 nM T83011 C6A8ZF 72696400 IC50 = 2980 nM T83011 C8ARZ1 72696401 IC50 > 10000 nM T83011 CB86ZM 72696517 IC50 = 1110 nM T83011 CH41BM 72696518 IC50 = 1160 nM T83011 CY9NX6 72696519 IC50 = 401 nM T83011 CQ4JZ3 72696520 IC50 > 10000 nM T83011 C4DN3V 72696521 IC50 = 3600 nM T83011 C4LCA1 72696649 IC50 = 518 nM T83011 CA71LP 72696650 IC50 = 437 nM T83011 C0R1CL 72696651 IC50 = 3430 nM T83011 CUY50L 72696652 IC50 = 1030 nM T83011 CU6RZ3 72696780 IC50 = 1240 nM T83011 CS5J3B 72696781 IC50 = 1090 nM T83011 CC4V8Y 72696782 IC50 = 15400 nM T83011 CIW4K9 72696784 IC50 = 2200 nM T83011 C1BDO7 72696917 IC50 = 1790 nM T83011 C1RE5Q 72696918 IC50 = 19730 nM T83011 CGP50Z 72696920 IC50 = 1360 nM T83011 CC2DB4 72697058 IC50 = 1560 nM T83011 CWG0U4 72697647 IC50 > 10000 nM T83011 CH90JS 72697648 IC50 > 10000 nM T83011 CPB7K4 72697649 IC50 = 10000 nM T83011 C1D7VQ 72697650 IC50 > 10000 nM T83011 C81TXZ 72697651 IC50 = 10000 nM T83011 CA5BI1 72697652 IC50 = 3760 nM T83011 C50SYX 72697785 IC50 = 1800 nM T83011 CXPB58 72697786 IC50 = 10000 nM T83011 CJ5W1R 72697787 IC50 = 10000 nM T83011 C0CJ6R 72697788 IC50 > 10000 nM T83011 CY1I8G 72697789 IC50 = 10000 nM T83011 CXDT98 72697790 IC50 > 10000 nM T83011 CS7VK8 72697791 IC50 > 10000 nM T83011 CX69MI 72697928 IC50 > 10000 nM T83011 CT2L7J 72697929 IC50 > 10000 nM T83011 CEWO96 72697930 IC50 > 10000 nM T83011 CNP9S3 72697931 IC50 > 10000 nM T83011 C3NR4V 72697932 IC50 > 10000 nM T83011 CQ4IE7 72697933 IC50 > 10000 nM T83011 CY94KO 72697934 IC50 > 10000 nM T83011 CO5K1Y 72698079 IC50 > 10000 nM T83011 CVB0Y9 72698080 IC50 = 10000 nM T83011 CCOP98 72698081 IC50 = 10000 nM T83011 C50ZUX 72698082 IC50 = 6390 nM T83011 CZG6V9 72698083 IC50 = 3260 nM T83011 C97FMG 72698084 IC50 > 10000 nM T83011 CH6Z2U 72698223 IC50 = 4760 nM T83011 C3QVP5 72698224 IC50 = 5870 nM T83011 CBD03K 72698225 IC50 > 10000 nM T83011 CST61L 72698226 IC50 = 3720 nM T83011 CJ0GB6 72698227 IC50 > 10000 nM T83011 CKP9M2 72698228 IC50 = 10000 nM T83011 C0WVR6 73334478 IC50 = 17000 nM T83011 CPFC15 73334583 IC50 = 5700 nM T83011 CS36LK 73334584 IC50 = 200 nM T83011 C81IEB 73334585 IC50 = 100 nM T83011 C04EOZ 73345930 IC50 = 42770 nM T83011 CL32OD 73346098 IC50 = 26.5 nM T83011 CT1NX3 73347452 IC50 = 18300 nM T83011 C3WZD5 73349093 IC50 = 13633 nM T83011 CQ0N6T 73352059 IC50 = 35860 nM T83011 C87CPY 73353370 IC50 = 185 nM T83011 C1L7MY 73353526 IC50 = 320 nM T83011 C5D4JS 73355020 IC50 = 16670 nM T83011 COJ7L5 73356449 IC50 = 24300 nM T83011 CPG73S 73417116 Ki = 26 nM T83011 CGD8R4 73671789 IC50 = 11800 nM T83011 C56INT 75395884 IC50 = 18.2 nM T83011 C74SVL 75414421 IC50 = 1462 nM T83011 C24XKD 76308234 IC50 = 79500 nM T83011 C68RKH 76310231 IC50 = 81000 nM T83011 CDK4R2 76310423 IC50 > 100000 nM T83011 CR1D2Z 76310442 IC50 = 7340 nM T83011 C3N5VB 76310836 IC50 = 31.5 nM T83011 C3XPT4 76310839 IC50 = 377 nM T83011 C9L3GR 76311136 IC50 > 100000 nM T83011 C5LW4R 76311137 IC50 = 15300 nM T83011 C7SX1Z 76311199 IC50 = 14210 nM T83011 CJ1W2I 76311204 IC50 = 34610 nM T83011 CL8N5U 76314097 IC50 > 100000 nM T83011 CJSF07 76314454 IC50 = 258 nM T83011 C8ZI4Y 76314455 IC50 = 82.4 nM T83011 CBKZ86 76314456 IC50 = 10000 nM T83011 CO8G2Y 76314457 IC50 = 0.588 nM T83011 CG70QL 76314458 IC50 = 120 nM T83011 C59NQU 76314463 IC50 = 13.5 nM T83011 C8FTG6 76314464 IC50 = 325 nM T83011 C1TFS4 76314802 IC50 = 7520 nM T83011 CM5I9G 76314803 IC50 = 92430 nM T83011 C2A8LT 76314813 IC50 > 100000 nM T83011 C59ZBF 76317227 IC50 = 452 nM T83011 CTX07R 76317228 IC50 = 257 nM T83011 CO1EN3 76317452 IC50 = 47000 nM T83011 CV6T1W 76317649 IC50 > 100000 nM T83011 CI9Z6N 76317651 IC50 > 100000 nM T83011 CC0B5D 76318043 IC50 = 1.41 nM T83011 CR45HD 76318044 IC50 = 123 nM T83011 CVDH35 76318045 IC50 = 41.7 nM T83011 CPB7I3 76318046 IC50 = 2.96 nM T83011 CKA48M 76318048 IC50 = 78.9 nM T83011 CY2QP8 76318337 IC50 = 150 nM T83011 CZ31JI 76318338 IC50 > 100000 nM T83011 CA5K6L 76318339 IC50 > 100000 nM T83011 CM97RB 76318340 IC50 > 100000 nM T83011 C38XFN 76318410 IC50 = 16290 nM T83011 C5JB3L 76318411 IC50 > 100000 nM T83011 CL4PU0 76318412 IC50 = 5010 nM T83011 C53ZLX 76318419 IC50 = 58310 nM T83011 C1C5FO 76318420 IC50 > 100000 nM T83011 CM54SP 76320939 IC50 = 440 nM T83011 C6XRT0 76321186 IC50 = 43300 nM T83011 C81DZU 76321374 IC50 > 100000 nM T83011 CSZ69D 76321757 IC50 = 52.6 nM T83011 CFD09Y 76321758 IC50 > 10000 nM T83011 CU5NB3 76321759 IC50 = 535 nM T83011 C0PW1A 76321760 IC50 > 10000 nM T83011 C84HGW 76321761 IC50 > 10000 nM T83011 CA3VD4 76321762 IC50 = 43.6 nM T83011 CSL45N 76321763 IC50 = 0.77 nM T83011 CC90FV 76322024 IC50 > 100000 nM T83011 CEI0B9 76322086 IC50 > 100000 nM T83011 CVXT29 76324406 Ki = 23000 nM T83011 CNS28Q 76324968 IC50 > 100000 nM T83011 C7VMB2 76324978 IC50 = 22300 nM T83011 CV29DJ 76325379 IC50 = 1440 nM T83011 CLU08E 76325380 IC50 > 10000 nM T83011 C7QV3I 76325640 IC50 > 100000 nM T83011 C0X6JA 76325641 IC50 = 100000 nM T83011 C2F4MQ 76325697 IC50 > 100000 nM T83011 CIT8F0 76325703 IC50 = 63770 nM T83011 C31JLR 76328918 IC50 = 24.7 nM T83011 CW14BN 76328919 IC50 = 2.62 nM T83011 CSR0P3 76328920 IC50 = 1.41 nM T83011 CERI13 76329220 IC50 = 100000 nM T83011 C0ED6S 76329275 IC50 = 40290 nM T83011 C5DS0O 76329943 IC50 = 54300 nM T83011 CDM84V 76332211 IC50 > 100000 nM T83011 CI8QE0 76332226 IC50 > 100000 nM T83011 CCR1U2 76332604 IC50 = 852 nM T83011 CUS43N 76332873 IC50 > 100000 nM T83011 CL4WZ8 76332874 IC50 > 100000 nM T83011 CW20MH 76332875 IC50 > 100000 nM T83011 CAEF41 76332923 IC50 = 12190 nM T83011 C91ENH 76332927 IC50 = 16190 nM T83011 C4PRU7 76332928 IC50 > 100000 nM T83011 C3B2GE 76334701 IC50 = 5940 nM T83011 C6XD0G 76335238 Ki = 9000 nM T83011 C67EJQ 76335845 IC50 = 62300 nM T83011 C2AEN5 76336201 IC50 = 67.1 nM T83011 CN0LI4 76336202 IC50 = 0.875 nM T83011 CG41IF 76336203 IC50 = 1790 nM T83011 CUNV46 76336531 IC50 = 97510 nM T83011 CH2T1L 76336532 IC50 = 10090 nM T83011 CKD2R8 76336533 IC50 = 14600 nM T83011 CD2J6U 76336534 IC50 = 89040 nM T83011 C0EXZ4 76336541 IC50 > 100000 nM T83011 C23YEG 76900387 IC50 = 6000 nM T83011 C9U8JP 77844601 Ki = 0.26 nM T83011 C3OP9Q 77844603 IC50 = 4.36 nM T83011 CH5YI4 77844667 Ki = 0.17 nM T83011 C83HNQ 77844716 Ki = 0.64 nM T83011 CYS0H9 77844719 Ki = 3.57 nM T83011 CL40EH 77844721 IC50 = 38.4 nM T83011 CU6K3W 77844723 Ki = 0.27 nM T83011 C9H7OG 77844769 Ki = 0.84 nM T83011 CUH8Z1 77844770 Ki = 0.93 nM T83011 C5VZ9M 77844771 Ki = 0.57 nM T83011 CR1Y5G 77844772 Ki = 0.46 nM T83011 CFWX23 82018566 IC50 > 10000 nM T83011 CQ1LF4 86043207 IC50 = 620 nM T83011 C1NI6G 86043210 IC50 = 1800 nM T83011 C0W2KN 86043213 IC50 = 3500 nM T83011 C7LDN8 86046220 IC50 = 59 nM T83011 C46NHO 86298552 IC50 = 4.5 nM T83011 C74WUO 86729878 IC50 = 32020 nM T83011 C4YE0G 87057445 IC50 > 1250000 nM T83011 CAE9S6 90197458 IC50 = 33300 nM T83011 C97DGB 90197459 IC50 = 190 nM T83011 CP4FQ2 90197685 IC50 = 5550 nM T83011 CB2RV3 90197737 IC50 = 28100 nM T83011 CJW98L 90197739 IC50 = 50500 nM T83011 C6AK9N 90197969 IC50 = 88 nM T83011 CS0ZH6 90197974 IC50 = 74300 nM T83011 CN7BV6 90479835 Ki = 0.5 nM T83011 CO51GW 90643508 IC50 = 10560 nM T83011 CB0AP6 90643928 IC50 = 6 nM T83011 C0QA7Z 90645389 IC50 = 10350 nM T83011 CF8T2J 90645390 IC50 = 45370 nM T83011 CG98IK 90645391 IC50 = 7410 nM T83011 CG1N2A 90645392 IC50 = 6500 nM T83011 C15POS 90645393 IC50 = 210 nM T83011 CD48PL 90645394 IC50 = 13090 nM T83011 CV42XE 90645395 IC50 = 7680 nM T83011 C6VL5U 90645396 IC50 = 16010 nM T83011 CY7C5S 90645397 IC50 = 25180 nM T83011 CO06VU 90645398 IC50 = 5680 nM T83011 CU5QE3 90645399 IC50 = 20710 nM T83011 CHDP57 90645400 IC50 = 15210 nM T83011 C9PIU7 90645500 IC50 = 111000 nM T83011 C8ZGF2 90645501 IC50 = 74500 nM T83011 CA8YH9 90645502 IC50 = 117000 nM T83011 CLJ8O4 90645503 IC50 = 224000 nM T83011 C8QI3X 90645505 IC50 = 215000 nM T83011 CR7UD8 90645506 IC50 = 100 nM T83011 C03REM 90646727 Ki = 1.45 nM T83011 C8RE0M 90646728 Ki = 4.82 nM T83011 CZF90P 90646729 Ki = 20.4 nM T83011 CV95XQ 90646731 Ki = 12.8 nM T83011 CV6X7K 90646732 Ki = 31.8 nM T83011 C8I7JS 90646833 Ki = 122 nM T83011 C40MQW 90656446 IC50 = 5.06 nM T83011 CF5I3K 90656447 IC50 = 9.34 nM T83011 C4P6YN 90656448 IC50 = 8.31 nM T83011 CRM6W2 90656449 IC50 = 38.03 nM T83011 C29OBX 90656450 IC50 = 65.49 nM T83011 C3JTI2 90656451 IC50 = 227.48 nM T83011 C7Y6XW 90656452 IC50 = 375.71 nM T83011 CNPR45 90656453 IC50 = 2.91 nM T83011 CI8AN7 90656454 IC50 = 9.13 nM T83011 C2DO3S 90656455 IC50 = 6.16 nM T83011 CX2BI1 90665464 IC50 = 3550 nM T83011 C2U4IX 90665465 IC50 = 3110 nM T83011 CRB45O 90665466 IC50 = 3560 nM T83011 C3FLR5 90665467 IC50 = 3940 nM T83011 CQB95X 90665468 IC50 = 15960 nM T83011 CV53TJ 90665469 IC50 = 3760 nM T83011 CX2J6R 90665471 IC50 = 2310 nM T83011 CY9HP0 90665472 IC50 = 2780 nM T83011 C1LYK6 90665473 IC50 = 8850 nM T83011 CVH28D 90665474 IC50 = 6000 nM T83011 C0BVY5 90665475 IC50 = 4780 nM T83011 CH8QE5 90665476 IC50 = 3750 nM T83011 C3VT2Z 90665477 IC50 = 2190 nM T83011 CDG71U 90665478 IC50 = 2880 nM T83011 COJ3I8 90665479 IC50 = 3490 nM T83011 CB2JY6 90665480 IC50 = 4530 nM T83011 CZ3K2I 90665481 IC50 = 10840 nM T83011 C98OBK 90665482 IC50 = 12610 nM T83011 CX1S7A 90665483 IC50 = 7550 nM T83011 CRLT57 90665484 IC50 = 1330 nM T83011 CR1IF2 90665485 IC50 = 2310 nM T83011 CUS3H7 90665486 IC50 = 1110 nM T83011 CZ2I3Q 90665487 IC50 = 2880 nM T83011 CXA4S3 90665488 IC50 = 1960 nM T83011 CQT26E 90665489 IC50 = 2310 nM T83011 C5LU6I 90665490 IC50 = 2290 nM T83011 CF4ZN3 90665491 IC50 = 4630 nM T83011 CAW89J 90665492 IC50 = 14530 nM T83011 C4YHG6 90665494 IC50 = 6230 nM T83011 CCEG94 90665495 IC50 = 4760 nM T83011 CBE9W8 90665496 IC50 = 7480 nM T83011 C1JCF4 90666201 IC50 = 22900 nM T83011 C0MNS2 90666203 IC50 = 10840 nM T83011 C53HVF 90666204 IC50 = 2100 nM T83011 C52ZRU 90666205 IC50 = 2340 nM T83011 CG7U0D 90666206 IC50 = 280 nM T83011 CEM2C7 90666207 IC50 = 6140 nM T83011 CFD4H5 90666208 IC50 = 880 nM T83011 C1YTP6 90666209 IC50 = 1370 nM T83011 C54YQR 90666210 IC50 = 6570 nM T83011 CHMD93 90666391 IC50 = 3020 nM T83011 CAS3P4 90667148 IC50 = 170 nM T83011 C9EDT4 90667149 IC50 = 30500 nM T83011 C14DIZ 90667150 IC50 = 72580 nM T83011 C1HJB5 90667151 IC50 = 5950 nM T83011 CIX7G5 90676868 IC50 = 716 nM T83011 C29MFT 90676892 IC50 = 393 nM T83011 CT15EF 91667541 IC50 = 6 nM T83011 C1SZM3 91809224 Ki = 60 nM T83011 C68YVN 91827407 IC50 > 200000 nM T83011 CZQ9E5 91863223 IC50 = 2.8 nM T83011 C90AXQ 91863224 IC50 = 1.3 nM T83011 C4GQ7A 91863375 IC50 = 13.25 nM T83011 CL45WP 91863383 IC50 = 52.93 nM T83011 C2XO9G 91973312 Ki = 16 nM T83011 CK59LE 91973747 IC50 = 74800 nM T83011 C58BTI 91973750 IC50 = 144 nM T83011 CF3I7E 96469773 IC50 = 8090 nM T83011 C9AG0E 101788293 IC50 = 21.35 nM T83011 C7H0SA 101788294 IC50 = 151.6 nM T83011 C08XPB 101896439 IC50 = 58910 nM T83011 C81WRJ 101910778 IC50 = 183.6 nM T83011 CQ1SM0 102004295 IC50 = 84600 nM T83011 C7CR9D 102220645 IC50 = 116 nM T83011 C3RW4H 102313434 IC50 > 100000 nM T83011 C0X7BR 107271816 IC50 = 2760 nM T83011 CR4W5N 110704124 IC50 = 141 nM T83011 CMY38C 112769743 IC50 = 10900 nM T83011 C9QS7H 112787413 IC50 = 14600 nM T83011 C4DAQ9 112788822 IC50 = 1690 nM T83011 CB2JW9 114940252 IC50 = 2.9 nM T83011 C8TX3R 115328020 IC50 = 20000 nM T83011 CQ8MX9 117929947 IC50 = 218 nM T83011 CKWG83 117939777 IC50 = 206 nM T83011 CL54XO 117939779 IC50 = 264 nM T83011 C4D5QS 117939782 IC50 = 22044 nM T83011 CP07SU 117939783 IC50 = 8000 nM T83011 CM8A4Q 117939786 IC50 = 911 nM T83011 CFYK36 117939787 IC50 = 894 nM T83011 C3JB9W 117939792 IC50 = 3749 nM T83011 CW7PI3 117939793 IC50 = 869 nM T83011 CE53IP 117939804 IC50 = 14086 nM T83011 C21BRF 117939805 IC50 = 26607 nM T83011 CMJF04 117939806 IC50 = 1260 nM T83011 C0HS3B 117939808 IC50 = 1380 nM T83011 CYW8F3 117939809 IC50 = 713 nM T83011 C7QP6F 117939810 IC50 = 21267 nM T83011 C76QNR 117939811 IC50 = 203 nM T83011 C75RLB 117939814 IC50 = 4372 nM T83011 C8W3YQ 117939815 IC50 = 7928 nM T83011 C4J5TP 117939817 IC50 = 864 nM T83011 CL30GA 117939818 IC50 = 532 nM T83011 CN6IS1 117939819 IC50 = 14219 nM T83011 CLU64K 117939825 IC50 = 1012 nM T83011 CW28FI 117939826 IC50 = 2109 nM T83011 CCS42Z 117945944 IC50 = 6400 nM T83011 CYBX18 118140875 IC50 = 280 nM T83011 C1J9DW 118140947 IC50 = 2500 nM T83011 CN7I8Q 118297734 IC50 > 200000 nM T83011 C61BNV 118304877 IC50 > 10000 nM T83011 C2U3NT 118483746 IC50 = 7 nM T83011 C38WNG 118483913 IC50 = 11500 nM T83011 C6A8FW 118483914 IC50 = 10400 nM T83011 CF7Z1S 118493308 IC50 > 10000 nM T83011 C10VNP 118536083 IC50 = 600 nM T83011 CF90SQ 118536088 IC50 = 62900 nM T83011 C9T8ZB 118536101 IC50 = 33000 nM T83011 C72EDN 118536105 IC50 > 100000 nM T83011 CYHM83 118536120 IC50 = 1600 nM T83011 C9BUT8 118536122 IC50 = 80200 nM T83011 CY2JZ4 118542609 IC50 = 24400 nM T83011 CC95BW 118706231 Ki = 980 nM T83011 CT1O7D 118706232 Ki = 700 nM T83011 CMS52X 118706233 Ki = 520 nM T83011 C3UE9R 118706234 Ki = 760 nM T83011 CUFL29 118706235 Ki = 990 nM T83011 C3M4SH 118706236 Ki = 1050 nM T83011 CY5DO8 118706237 Ki = 870 nM T83011 C4VA3Z 118706239 Ki = 900 nM T83011 C3AY6U 118709465 IC50 = 220 nM T83011 C87JAX 118709466 IC50 > 10000 nM T83011 CCH7X5 118709467 IC50 = 388 nM T83011 C1BF7M 118709468 IC50 > 10000 nM T83011 CU2Y0H 118709469 IC50 = 2270 nM T83011 C4H1TQ 118712953 IC50 = 600 nM T83011 C4J8TS 118712954 IC50 = 12700 nM T83011 CH0YP2 118712955 IC50 = 941 nM T83011 C2BZ4I 118712956 IC50 = 998 nM T83011 CR34TU 118718853 IC50 = 5.32 nM T83011 COG7T6 118720585 IC50 = 330 nM T83011 CS5HX1 118720586 IC50 = 120 nM T83011 CKV3E8 118720587 IC50 = 110 nM T83011 CQ05ZR 118724437 IC50 = 5520 nM T83011 CX93MC 118724438 IC50 = 2.1 nM T83011 C3KEL9 118724439 IC50 = 2170 nM T83011 CM5J3R 118724440 IC50 = 2.2 nM T83011 C5IN1P 118724441 IC50 = 4.1 nM T83011 C57BEW 118726138 IC50 = 52880 nM T83011 C2UX0J 118726140 IC50 = 59400 nM T83011 C1WGY9 118726141 IC50 = 45610 nM T83011 C7GXD9 118726142 IC50 = 50580 nM T83011 CZ28ED 118726143 IC50 = 47360 nM T83011 C3A2XO 118726144 IC50 = 40090 nM T83011 C1IBC8 118726146 IC50 = 56210 nM T83011 CDX5V0 118726148 IC50 = 44090 nM T83011 CC87QU 118726153 IC50 = 31550 nM T83011 CTBQ68 118726154 IC50 = 56500 nM T83011 CZ8DR0 118726156 IC50 = 30170 nM T83011 C8PRQ1 118726157 IC50 = 55100 nM T83011 C05AKN 118726159 IC50 = 41320 nM T83011 CDX2G5 118726160 IC50 = 59400 nM T83011 CC4R5P 118726163 IC50 = 16090 nM T83011 C3COH5 118726165 IC50 = 55850 nM T83011 CN4GY5 118726166 IC50 = 41800 nM T83011 CIZ8P9 118726168 IC50 = 49890 nM T83011 CO3N6F 118726169 IC50 = 58940 nM T83011 CSJR39 118726170 IC50 = 42320 nM T83011 C17VOQ 118726172 IC50 = 30080 nM T83011 C37VRU 118726187 IC50 = 413 nM T83011 CRJD86 118726188 IC50 = 542 nM T83011 C2TU4X 118726189 IC50 = 1236 nM T83011 C80FUE 118726190 IC50 = 9334 nM T83011 C4VX5E 118727528 IC50 > 100000 nM T83011 C1LK6U 118727529 IC50 > 100000 nM T83011 C6PX9T 118727530 IC50 > 100000 nM T83011 C3HD8M 118727531 IC50 = 11900 nM T83011 CADH94 118727532 IC50 = 1520 nM T83011 C9G1YD 118727533 IC50 = 2860 nM T83011 CRN59D 118727534 IC50 > 100000 nM T83011 CTH6S4 118727535 IC50 = 20 nM T83011 CY8Q9V 118727536 IC50 = 1270 nM T83011 CP7A9D 118727537 IC50 > 100000 nM T83011 CFWJ56 118728390 IC50 = 36000 nM T83011 CMEA81 118728391 IC50 = 27000 nM T83011 CJ8ZY2 118728392 IC50 = 19000 nM T83011 CW8Z2H 118728853 IC50 > 100000 nM T83011 C9XEY8 118728854 IC50 > 100000 nM T83011 CVCT10 118728855 IC50 > 100000 nM T83011 C1JX3S 118728856 IC50 > 100000 nM T83011 CULF09 118728857 IC50 > 100000 nM T83011 CDKA92 118728858 IC50 > 100000 nM T83011 C4XUG3 118728859 IC50 > 100000 nM T83011 CK3E9J 118728860 IC50 > 100000 nM T83011 C8L6TZ 118728861 IC50 > 100000 nM T83011 CS8UI6 118728862 IC50 > 100000 nM T83011 CAZ78X 118728978 IC50 = 3310 nM T83011 CXG4B7 118728979 IC50 = 7290 nM T83011 C7UED4 118728980 IC50 = 168 nM T83011 CK9AX4 118728981 IC50 = 57 nM T83011 C68EHZ 118728982 Ki = 41 nM T83011 C1LY8F 118728983 IC50 = 48 nM T83011 CVP9F5 118728984 IC50 = 947 nM T83011 C6HFT1 118728985 IC50 = 348 nM T83011 CUZ96B 118728986 IC50 = 941 nM T83011 CW65QL 118729284 IC50 = 8300 nM T83011 CXOA52 118730192 IC50 = 196.3 nM T83011 C27ZWI 118730193 IC50 = 35100 nM T83011 CEQ56Z 118730194 IC50 = 33600 nM T83011 C3D6VY 118730195 IC50 = 21300 nM T83011 CJ2P9D 118730196 IC50 = 1000 nM T83011 CI2X8N 118730197 IC50 = 13500 nM T83011 CP70TH 118730198 IC50 = 7900 nM T83011 CPAT89 118730199 IC50 = 164700 nM T83011 C5F4LP 118730200 IC50 = 273100 nM T83011 C07UCB 118733540 IC50 = 60 nM T83011 CM76SB 118733551 IC50 = 56 nM T83011 C6RY3J 118734094 IC50 = 12290 nM T83011 C0SR8X 118734098 IC50 = 84700 nM T83011 C0J2WE 118734102 IC50 = 19170 nM T83011 CW81OF 118734104 IC50 = 21200 nM T83011 CH7OT9 118734108 IC50 = 80070 nM T83011 C3XB0N 118734706 IC50 = 1520 nM T83011 CK4C6E 118734707 IC50 = 37960 nM T83011 C0S9TQ 118734709 IC50 = 28760 nM T83011 C67ZXU 118734710 IC50 = 25730 nM T83011 CR28OT 118734711 IC50 = 5770 nM T83011 CNB83Q 118734712 IC50 = 700 nM T83011 CX80VO 118734713 IC50 = 240 nM T83011 CB87ZI 118734714 IC50 = 540 nM T83011 CDO43K 118734715 IC50 = 1770 nM T83011 C67CLN 118734716 IC50 = 9510 nM T83011 C5SN4X 118734717 IC50 = 2290 nM T83011 CI71ZY 118734718 IC50 = 3450 nM T83011 CIC36U 118734719 IC50 = 2260 nM T83011 C1R8IE 118734720 IC50 = 2000 nM T83011 CSDJ67 118734721 IC50 = 5280 nM T83011 CN3S6M 118734722 IC50 = 1590 nM T83011 C71YMX 118734723 IC50 = 780 nM T83011 C89PQZ 118734724 IC50 = 2370 nM T83011 CWR41B 118734725 IC50 = 4560 nM T83011 C7Y0LX 118735096 IC50 = 42650 nM T83011 C41EPX 118913669 IC50 = 7600 nM T83011 CJ5NC9 118913682 IC50 = 7160 nM T83011 C1ENW9 118913743 IC50 > 100000 nM T83011 CQNM60 118918087 IC50 > 100000 nM T83011 CGZ1L3 118931167 IC50 > 100000 nM T83011 CMX4J6 121482363 IC50 = 360579 nM T83011 CD9H0B 122179917 IC50 = 310 nM T83011 C9P1NG 122179918 IC50 = 520 nM T83011 CK3T9I 122179919 IC50 = 210 nM T83011 C6RZ5L 122179920 IC50 > 1000 nM T83011 C4U0ER 122179921 IC50 > 1000 nM T83011 C3ZST9 122179922 IC50 = 310 nM T83011 CC41ST 122179923 IC50 > 1000 nM T83011 C6EZH1 122179924 IC50 = 310 nM T83011 C4ENL2 122179925 IC50 > 1000 nM T83011 CO8K2X 122179926 IC50 = 950 nM T83011 C6C5YK 122179927 IC50 = 430 nM T83011 CM5R7F 122180400 IC50 = 134 nM T83011 C6PTD5 122180404 IC50 = 96 nM T83011 C1X9KB 122180406 IC50 = 29 nM T83011 CMC26Y 122180416 IC50 = 321 nM T83011 C8UIY9 122180417 IC50 = 18 nM T83011 CEJ8S0 122180431 IC50 = 41 nM T83011 CJK24Z 122180436 IC50 = 53 nM T83011 C3ZJF5 122180450 IC50 = 45 nM T83011 C7IFX2 122180453 IC50 = 17 nM T83011 C5LT1G 122180455 IC50 = 39 nM T83011 CTO9N3 122180457 IC50 = 24 nM T83011 CKM1E7 122180462 IC50 = 10 nM T83011 CMD2B6 122180465 IC50 = 24 nM T83011 C79SBR 122180468 IC50 = 5.7 nM T83011 CV48UD 122185513 Ki = 22 nM T83011 C30IGS 122185514 Ki = 22000 nM T83011 CM2PD5 122186418 IC50 = 7100 nM T83011 C1V5AO 122186419 IC50 = 1600 nM T83011 CQ5PO2 122186420 IC50 = 14200 nM T83011 CD0V5N 122186421 IC50 = 3900 nM T83011 C4L3WE 122186422 IC50 = 360 nM T83011 C21HOI 122186423 IC50 = 97 nM T83011 CH35KZ 122186425 IC50 = 51 nM T83011 C03TJD 122186427 IC50 = 66 nM T83011 CEVY24 122186429 IC50 = 60 nM T83011 CC91RU 122186431 IC50 = 5100 nM T83011 CO0B7A 122186433 IC50 = 2900 nM T83011 CM94AW 122186435 IC50 = 23100 nM T83011 CA4M3I 122186437 IC50 = 20800 nM T83011 C8YIT5 122186439 IC50 = 320 nM T83011 C2PC4U 122186440 IC50 = 650 nM T83011 CZS2M9 122186441 IC50 = 690 nM T83011 C5VNO0 122186442 IC50 = 3900 nM T83011 CZ5B7W 122186443 IC50 = 9800 nM T83011 CA4GO3 122188866 IC50 > 10000 nM T83011 CNYA71 122188867 IC50 > 10000 nM T83011 CCEQ57 122188868 IC50 = 5980 nM T83011 CHK2M9 122188869 IC50 = 3370 nM T83011 C5SNF1 122188870 IC50 = 5880 nM T83011 C1K0PT 122188871 IC50 = 2590 nM T83011 COM53A 122194326 IC50 = 9170 nM T83011 C2E6HQ 122194327 IC50 = 22350 nM T83011 C05DBN 122194328 IC50 = 4200 nM T83011 CYHF09 122194329 IC50 > 60000 nM T83011 C16GMN 122194330 IC50 = 14500 nM T83011 CS1UH0 122194331 IC50 = 20010 nM T83011 CN9CU1 122194332 IC50 = 2780 nM T83011 CTED74 122194333 IC50 = 5090 nM T83011 C8ZPO0 122194334 IC50 = 10160 nM T83011 C0B7ED 122194335 IC50 = 7360 nM T83011 CI9F4S 122194603 IC50 > 60000 nM T83011 C4MQP9 122194604 IC50 > 60000 nM T83011 CU1HE5 122194605 IC50 = 55300 nM T83011 CV5RC2 122194606 IC50 > 60000 nM T83011 C4OEV3 122194607 IC50 > 60000 nM T83011 CR62NI 122194608 IC50 = 48090 nM T83011 C8VQA9 122194609 IC50 = 35500 nM T83011 CHRQ34 122194610 IC50 > 60000 nM T83011 CSZ72C 122194611 IC50 = 50520 nM T83011 CLZ8S5 122194612 IC50 > 60000 nM T83011 CA79DS 122415289 IC50 > 50000 nM T83011 C9U0EL 124115926 IC50 = 966 nM T83011 C5WHS1 124116114 IC50 = 2740 nM T83011 CR81DC 124116115 IC50 = 13 nM T83011 C01TOU 124116118 IC50 = 30 nM T83011 C8U5RC 124313549 IC50 = 100000 nM T83011 CI5M3O 126842840 IC50 = 2680 nM T83011 CO01UP 127025001 IC50 = 23400 nM T83011 CT6H9W 127025002 IC50 = 14700 nM T83011 C6N1OH 127025105 IC50 = 2878 nM T83011 CP5VQ6 127025106 IC50 = 3522 nM T83011 CW7U0M 127025386 IC50 = 2568 nM T83011 C32MKJ 127025613 IC50 = 8390 nM T83011 CK28JE 127025614 IC50 = 12600 nM T83011 CS3UX1 127025615 IC50 = 30400 nM T83011 CMI23B 127025616 IC50 = 2750 nM T83011 C8HT6M 127025617 IC50 = 33900 nM T83011 C21OBG 127025662 IC50 = 504 nM T83011 CRQS79 127025663 IC50 = 584 nM T83011 C9H5EW 127025664 IC50 = 467 nM T83011 C65JIY 127025665 IC50 = 45240 nM T83011 CTR92D 127025666 IC50 = 34670 nM T83011 C1XI6Y 127025668 IC50 = 452 nM T83011 CL3RP0 127025669 IC50 = 348 nM T83011 CZ9CJ8 127025670 IC50 = 221 nM T83011 C5O8ZV 127025898 IC50 = 33600 nM T83011 CJRV60 127025899 IC50 = 31900 nM T83011 CH6A2X 127026192 IC50 = 2620 nM T83011 C2MHZ4 127026193 IC50 = 40500 nM T83011 C6GNR7 127026321 IC50 = 1321 nM T83011 CSAJ72 127026323 IC50 = 2722 nM T83011 CN0A5U 127026324 IC50 = 1634 nM T83011 C0MDO2 127026857 IC50 = 1782 nM T83011 CNR05U 127027039 Ki = 9700 nM T83011 C8WJF6 127027348 Ki = 18700 nM T83011 C8WB9H 127027461 IC50 = 523.46 nM T83011 C0Y8QM 127027785 IC50 = 9.46 nM T83011 CT6AD7 127027787 IC50 = 242 nM T83011 C5A9ZJ 127028005 Ki = 2600 nM T83011 CXSK51 127028089 IC50 = 626.82 nM T83011 C9XRA0 127028155 IC50 = 84.1 nM T83011 C5IGO0 127028297 Ki = 10600 nM T83011 C4FZ7Y 127029319 IC50 = 19.35 nM T83011 C0MTE2 127029587 IC50 = 217.99 nM T83011 C57BAC 127029589 IC50 = 67.69 nM T83011 CX53RY 127029592 IC50 = 2460 nM T83011 CL15QN 127029593 IC50 = 203.59 nM T83011 C18CJS 127029594 IC50 = 7.61 nM T83011 C19THR 127030340 IC50 = 334 nM T83011 CKHY89 127031268 IC50 = 703 nM T83011 CDL0C7 127031303 IC50 > 100000 nM T83011 CLT4M1 127031655 IC50 = 87 nM T83011 C6AI2K 127031680 Ki = 1150 nM T83011 CJ2U6F 127032119 IC50 = 391 nM T83011 C0C9WI 127032253 IC50 > 100000 nM T83011 C9W3MT 127033454 IC50 = 1510 nM T83011 C8FIK0 127034240 IC50 = 10800 nM T83011 C4B2YX 127034243 IC50 = 1500 nM T83011 C0RB9X 127034301 Ki = 720 nM T83011 CQT5M1 127034333 IC50 = 27800 nM T83011 COY03I 127034334 IC50 > 100000 nM T83011 CMR83A 127034503 IC50 = 226 nM T83011 C69KJB 127034561 IC50 = 808 nM T83011 CAH75M 127034731 IC50 = 174.8 nM T83011 C9RB7W 127035092 IC50 = 3760 nM T83011 C94YFD 127035093 IC50 = 2580 nM T83011 CGDB19 127035094 IC50 = 5670 nM T83011 C8K1NG 127035095 IC50 = 60.1 nM T83011 C6KME4 127035096 IC50 = 401.3 nM T83011 C3LJ9W 127035097 IC50 = 2450 nM T83011 CG5SI3 127035266 IC50 = 330 nM T83011 CIP89M 127035390 IC50 = 218 nM T83011 C06VIZ 127035396 IC50 = 256.4 nM T83011 CW2XJ0 127035397 IC50 = 201 nM T83011 CA08TK 127035398 IC50 = 105.6 nM T83011 CR4WJ7 127035399 IC50 = 253.2 nM T83011 CC45DE 127035495 IC50 = 75800 nM T83011 C9SEO1 127035497 IC50 = 3900 nM T83011 CN1JC8 127035507 IC50 > 60000 nM T83011 C2DL5A 127035509 IC50 > 70000 nM T83011 C9GMF4 127035552 IC50 = 904.6 nM T83011 C5PH0B 127035553 IC50 = 305.2 nM T83011 CMP1D6 127035554 IC50 = 651.1 nM T83011 C4AD2V 127035673 IC50 = 4430 nM T83011 CG70KY 127035960 IC50 = 830 nM T83011 C1XAW5 127035961 IC50 = 1400 nM T83011 CB5W1U 127035962 IC50 = 185 nM T83011 CS4B8G 127036275 IC50 = 3670 nM T83011 C5SUJ2 127036479 IC50 = 1130 nM T83011 CUZR67 127036672 IC50 = 67 nM T83011 CWDI07 127037076 IC50 = 3270 nM T83011 CY7AX6 127037276 IC50 = 938.4 nM T83011 C81AIF 127037457 IC50 = 714.1 nM T83011 CL29WO 127037458 IC50 = 803 nM T83011 C0S8GJ 127037470 IC50 = 10710 nM T83011 C7F6UN 127037705 IC50 = 127150 nM T83011 C5MRS1 127037706 IC50 = 83060 nM T83011 C2W4DY 127037999 IC50 = 112130 nM T83011 C9HIT0 127038000 IC50 = 98.32 nM T83011 C9TC4Q 127038068 IC50 = 110650 nM T83011 C96BZR 127038887 IC50 = 1930 nM T83011 CN3QG5 127038898 IC50 = 33 nM T83011 CI9VS5 127039241 IC50 = 28500 nM T83011 CWS57M 127039242 IC50 = 45600 nM T83011 C7OES9 127039243 IC50 = 2380 nM T83011 CV03PG 127039401 IC50 = 91.29 nM T83011 CS8G3X 127039402 IC50 = 55.37 nM T83011 CB9IX7 127041996 IC50 = 251.14 nM T83011 C0V5DN 127041997 IC50 = 21450 nM T83011 C3C4UD 127042054 IC50 = 69560 nM T83011 C54KZB 127042056 IC50 = 167980 nM T83011 C9US1F 127042057 IC50 = 100020 nM T83011 CLX9A4 127042315 IC50 = 52.23 nM T83011 CSD84W 127042330 IC50 = 58.82 nM T83011 C1NB5G 127042331 IC50 = 33.45 nM T83011 CL5OX4 127042332 IC50 = 30.27 nM T83011 CRJE48 127042333 IC50 = 21.56 nM T83011 C82PWS 127042399 IC50 = 108090 nM T83011 CNI8Z2 127042400 IC50 = 107310 nM T83011 CF7BE1 127042742 IC50 = 90880 nM T83011 CKS6M1 127042743 IC50 = 153070 nM T83011 CN6HZ3 127042941 IC50 = 3 nM T83011 C3Z8FA 127042942 IC50 = 5 nM T83011 CU04BL 127042970 IC50 = 47.28 nM T83011 CN46BI 127043830 IC50 > 10000 nM T83011 CJ6W2U 127045743 IC50 = 10300 nM T83011 CGUC67 127045964 IC50 > 100000 nM T83011 C4DRT5 127046073 IC50 > 100000 nM T83011 CT0DZ1 127046074 IC50 > 100000 nM T83011 CXP8S3 127046075 IC50 > 100000 nM T83011 C71PDE 127046206 IC50 > 100000 nM T83011 C5KOC8 127046207 IC50 > 100000 nM T83011 C4MOG6 127046208 IC50 > 100000 nM T83011 CTDZ75 127046395 IC50 > 100000 nM T83011 CTVO57 127046396 IC50 = 581 nM T83011 CG8X9O 127046431 IC50 > 100000 nM T83011 CW51KH 127046559 IC50 > 100000 nM T83011 C5P7UB 127046560 IC50 > 100000 nM T83011 CI7AO8 127046561 IC50 > 100000 nM T83011 CYNG69 127046593 IC50 > 100000 nM T83011 CH4MZ0 127046738 IC50 = 7460 nM T83011 CIK0O4 127046739 IC50 = 1940 nM T83011 C3H2TR 127046740 IC50 = 56200 nM T83011 C75RDT 127046765 IC50 = 923 nM T83011 CC14IO 127047102 IC50 > 100000 nM T83011 CHQ3V7 127047235 IC50 > 100000 nM T83011 CC4R1Z 127047236 IC50 = 6790 nM T83011 C90YDX 127047237 IC50 = 1210 nM T83011 CREG96 127047238 IC50 > 100000 nM T83011 CU39GI 127047239 IC50 > 100000 nM T83011 CN46VR 127047342 IC50 = 83100 nM T83011 CCS71F 127047626 IC50 > 100000 nM T83011 CW7A9C 127047746 IC50 = 3750 nM T83011 CZ1L4H 127047856 IC50 > 100000 nM T83011 C9EML8 127047875 IC50 > 100000 nM T83011 C8V2DN 127048404 IC50 > 100000 nM T83011 CW2B3M 127048716 IC50 > 100000 nM T83011 CZ2U0R 127048829 IC50 = 10.58 nM T83011 C23EOB 127049071 IC50 = 6000 nM T83011 CU85GC 127049730 IC50 = 13100 nM T83011 C31KDR 127050122 IC50 = 241.11 nM T83011 CH42VA 127050173 IC50 = 10620 nM T83011 CSJX42 127050454 IC50 = 18330 nM T83011 C0I4EF 127051346 IC50 = 2390 nM T83011 CD3Z8O 127051347 IC50 = 213.22 nM T83011 C12ZWP 127051348 IC50 = 10510 nM T83011 C8P5WZ 127051349 IC50 = 13760 nM T83011 CS78CM 127051350 IC50 = 10210 nM T83011 C71ZRS 127052872 IC50 = 10400 nM T83011 C83LIY 129165316 IC50 > 10000 nM T83011 CJGE94 129165458 IC50 > 10000 nM T83011 C84UJE 130302628 IC50 > 30000 nM T83011 C3M2IV 130344977 IC50 = 16400 nM T83011 CE8Q7I 130345035 IC50 > 100000 nM T83011 C01UGK 130345060 IC50 = 46200 nM T83011 CN9S7B 130345097 IC50 > 100000 nM T83011 C3CH7B 130345110 IC50 > 100000 nM T83011 C7RN8L 130345158 IC50 > 100000 nM T83011 CF20BS 130345178 IC50 > 100000 nM T83011 CMO50A 130345200 IC50 = 87000 nM T83011 C29WVS 130358344 IC50 > 100000 nM T83011 CZM13E 130358354 IC50 > 100000 nM T83011 CW47IH 130638185 IC50 = 40900 nM T83011 CP8L7V 132137973 IC50 > 100000 nM T83011 CRG1Y4 132342060 IC50 > 100000 nM T83011 CZ3OD0 132495360 IC50 = 53904 nM T83011 CBN5C0 132495361 IC50 > 100000 nM T83011 CWO31Y 132495367 IC50 = 1740 nM T83011 C2CJF3 132503347 IC50 = 816 nM T83011 C7DC2X 132511215 IC50 > 100000 nM T83011 C0ERW7 132511218 IC50 > 100000 nM T83011 CL9UY5 132511220 IC50 > 100000 nM T83011 CL23KG 132571526 IC50 = 2420 nM T83011 CO8P7W 132576240 IC50 = 143.65 nM T83011 CF3X5S 132577022 IC50 = 129000 nM T83011 C1TJ7B 132578491 IC50 > 10000 nM T83011 C5CKG0 132578492 IC50 = 210 nM T83011 CVS8H1 132578493 IC50 > 10000 nM T83011 CYB73H 132579936 IC50 = 11200 nM T83011 CF3M0N 132579937 IC50 = 3500 nM T83011 C9MRW2 132579938 IC50 = 600 nM T83011 CGIQ08 132579939 IC50 = 5200 nM T83011 CV7IT1 132819950 IC50 = 290 nM T83011 CTQ51R 132938089 IC50 > 1000 nM T83011 C61OMY 132941420 IC50 = 0.4 nM T83011 C4SOK7 132941421 Ki = 0.31 nM T83011 C87SOL 132961376 IC50 = 900 nM T83011 C6U1LV 132969040 IC50 > 100000 nM T83011 C45WQG 132969041 Ki = 3580 nM T83011 CL6XW8 132969042 Ki = 2570 nM T83011 C94JLM 133053560 Ki = 31 nM T83011 C1A7TX 134130045 IC50 = 710 nM T83011 CM23HY 134130366 IC50 = 6700 nM T83011 C71LDW 134130716 IC50 = 780 nM T83011 CR7M3J 134130929 IC50 = 710 nM T83011 CMC8D2 134131068 IC50 = 2100 nM T83011 C6WY4Q 134131214 IC50 = 3500 nM T83011 CF4OX9 134131513 IC50 = 2480 nM T83011 CBJ3G2 134131700 IC50 = 13.87 nM T83011 CCJF74 134132255 IC50 > 100000 nM T83011 CG1TY4 134132538 IC50 = 215 nM T83011 CRY9P0 134133186 IC50 = 316 nM T83011 CHT37D 134133216 IC50 = 376 nM T83011 C6VS5U 134133379 IC50 > 100000 nM T83011 CVF3T5 134133384 IC50 > 100000 nM T83011 CK3BW5 134134850 IC50 = 1010 nM T83011 CFQN14 134135653 IC50 = 14000 nM T83011 CP3RN6 134136543 IC50 > 100000 nM T83011 CSA09I 134137557 IC50 > 100000 nM T83011 C97CUD 134137716 IC50 > 100000 nM T83011 CV3J2Q 134138913 IC50 = 47 nM T83011 CF76XM 134139033 IC50 = 8.35 nM T83011 CQU8T5 134139124 IC50 > 100000 nM T83011 CJ6AO0 134139236 IC50 > 100000 nM T83011 C51HUD 134140107 Ki = 55180 nM T83011 CF9C1X 134140379 IC50 = 471 nM T83011 C73LGF 134140781 IC50 > 100000 nM T83011 CV60BZ 134140877 IC50 = 882 nM T83011 CFJ74X 134140944 IC50 = 14 nM T83011 C5ZD3G 134142101 IC50 = 1340 nM T83011 CB6FU0 134142341 IC50 = 1150 nM T83011 CSYM31 134142478 IC50 = 59293 nM T83011 CKD8B9 134142584 IC50 = 722 nM T83011 CUP09Q 134142596 IC50 > 100000 nM T83011 C0S6OI 134142875 Ki = 30380 nM T83011 CDGY36 134144163 IC50 = 1500 nM T83011 C47KWL 134144584 IC50 > 100000 nM T83011 C0HDQ1 134144802 IC50 = 2430 nM T83011 CP0D4F 134146126 IC50 > 100000 nM T83011 CZM9O4 134146757 IC50 = 7700 nM T83011 C3RHY4 134147228 IC50 = 5.3 nM T83011 C7E3YA 134149382 IC50 > 100000 nM T83011 C0V3GR 134149702 IC50 = 6.41 nM T83011 CJ1D3P 134149885 IC50 = 84 nM T83011 C4Y5ZX 134150471 IC50 = 8300 nM T83011 CRZ2W4 134150858 IC50 > 100000 nM T83011 C8XJH0 134151923 IC50 = 13 nM T83011 C83ZAR 134152670 IC50 = 915 nM T83011 CJ98WY 134152913 IC50 > 100000 nM T83011 CF8RV4 134153109 IC50 = 130 nM T83011 CA2KR0 134153338 IC50 > 100000 nM T83011 CPBG73 134153558 IC50 > 100000 nM T83011 C95UFC 134154267 IC50 = 29000 nM T83011 CGK4X3 134155114 IC50 = 52 nM T83011 C9QXG2 134155279 IC50 > 100000 nM T83011 C0IVJ4 134155685 IC50 = 190 nM T83011 CQA14Y 134155772 IC50 > 100000 nM T83011 C07ZGI 134156270 IC50 = 5.2 nM T83011 C4LW3F 134156704 IC50 = 1720 nM T83011 C9A2GK 134156912 IC50 > 100000 nM T83011 CC0IG7 134157232 IC50 = 72611 nM T83011 CWRT82 134157848 IC50 = 1030 nM T83011 CK1C8S 134366896 IC50 = 3363.5 nM T83011 CES20P 134366906 IC50 = 370.1 nM T83011 C7G9XA 134366910 IC50 = 38.1 nM T83011 C1HKG7 134366921 IC50 = 7440.7 nM T83011 C67XBZ 134366929 IC50 = 14159.5 nM T83011 C5TES6 134366930 IC50 = 4603.4 nM T83011 C5BKG0 134366932 IC50 = 216.4 nM T83011 C6X3EJ 134366939 IC50 = 501.8 nM T83011 CX8UB1 134366949 IC50 = 10.9 nM T83011 CD0B8J 134366950 IC50 = 57 nM T83011 CNC96K 134366956 IC50 = 5554.5 nM T83011 CK05MI 134366959 IC50 = 159 nM T83011 CCX21V 134366961 IC50 = 7 nM T83011 CQ80YU 134366964 IC50 = 67 nM T83011 C59ORQ 134366996 IC50 = 56.6 nM T83011 C1U7QY 134385634 IC50 = 436.2 nM T83011 CL0QX6 134385635 IC50 = 21.2 nM T83011 C83FUK 134385636 IC50 = 5048.7 nM T83011 C1APN4 134385637 IC50 = 147 nM T83011 C0CU9Q 134385638 IC50 = 417.6 nM T83011 CFU6H7 134385639 IC50 = 342.2 nM T83011 CP8VX4 134385640 IC50 = 3540.2 nM T83011 CL18CZ 134385641 IC50 = 68.1 nM T83011 C2ZGM9 134385642 IC50 = 1737 nM T83011 CX2I7K 134385643 IC50 = 549.7 nM T83011 C6HB5G 134385645 IC50 = 11830.4 nM T83011 C74VGX 134385646 IC50 = 18.6 nM T83011 C9QZH6 134385648 IC50 = 44.4 nM T83011 CK6L7Y 134385649 IC50 = 43.7 nM T83011 CL4UG2 134385650 IC50 = 50.4 nM T83011 C9LNR7 134816193 IC50 = 0.8 nM T83011 CA2H1G 134816270 IC50 = 1700 nM T83011 CEYR15 134816271 IC50 = 300 nM T83011 CTOB53 134816331 IC50 = 530 nM T83011 C2X3GF 134816595 IC50 = 470 nM T83011 CD9B4Z 134816640 IC50 = 1550 nM T83011 C35ZVJ 134816641 IC50 = 1.3 nM T83011 C4R6KL 134816691 IC50 = 3600 nM T83011 C0IOP2 134816692 IC50 = 1410 nM T83011 CC94YQ 134816693 IC50 = 290 nM T83011 CP86GA 134816695 IC50 = 5640 nM T83011 CUD08L 134817200 IC50 = 78 nM T83011 C2ATF7 135401432 IC50 = 59333 nM T83011 CH4L1K 135408573 IC50 = 3030 nM T83011 C0UCX3 135408731 IC50 > 10000 nM T83011 CRS0F8 135412828 IC50 = 60 nM T83011 C84CMF 135417113 IC50 = 1240 nM T83011 C14TDX 135418929 IC50 = 2500 nM T83011 CR1LE3 135432900 Ki = 38 nM T83011 CYW76V 135433346 IC50 = 482 nM T83011 C5T9YE 135436602 IC50 = 120000 nM T83011 CNQ3D5 135438796 IC50 = 31800 nM T83011 C1DKU8 135441424 IC50 = 230 nM T83011 C8WL0I 135449090 IC50 = 9017 nM T83011 CSW7P4 135454250 IC50 = 42.3 nM T83011 C2WA9R 135457295 IC50 = 100000 nM T83011 CGFS08 135459067 IC50 = 13320 nM T83011 CTE23K 135464118 IC50 = 11333 nM T83011 CB53EI 135465870 IC50 = 33833 nM T83011 CA07BI 135465901 Ki = 30 nM T83011 CHNA50 135471217 IC50 = 20000 nM T83011 C7AGR0 135474338 IC50 = 3800 nM T83011 CJR38B 135483618 IC50 = 19000 nM T83011 CKG25Y 135495099 IC50 = 7200 nM T83011 CT3M5A 135497038 IC50 = 25000 nM T83011 CCDS87 135499808 IC50 = 89000 nM T83011 C34FXW 135501716 IC50 = 2567 nM T83011 CHGR35 135505744 IC50 = 3000 nM T83011 CCJA58 135509938 IC50 = 30000 nM T83011 C6VS7P 135514579 IC50 = 30000 nM T83011 C1CZ9M 135514796 IC50 = 33000 nM T83011 CR05TL 135516788 IC50 = 130000 nM T83011 CD2X0Y 135524872 IC50 = 42000 nM T83011 COKH19 135526739 IC50 = 566 nM T83011 C3G2MZ 135538313 IC50 = 779 nM T83011 C0H8ZL 135657342 IC50 = 25130 nM T83011 CIAN64 135657390 IC50 = 31740 nM T83011 CJ5HX4 135657424 IC50 = 6500 nM T83011 CY57UW 135719318 IC50 = 1400 nM T83011 C60MRN 135719324 IC50 = 5990 nM T83011 CCNH91 135743577 IC50 > 300000 nM T83011 CZ97SK 135778696 IC50 = 1300 nM T83011 C06ZWB 135787694 IC50 = 60930 nM T83011 CBN2V5 135787695 IC50 = 10710 nM T83011 C03HVY 135846955 IC50 = 34333 nM T83011 CQCT18 135846958 IC50 = 35667 nM T83011 CE4QG5 135846981 IC50 = 30467 nM T83011 C3UB7L 135846982 IC50 = 25733 nM T83011 CON48D 135860273 IC50 = 69380 nM T83011 CQ24GS 135888977 IC50 = 723 nM T83011 CKDW41 135966009 IC50 = 24333 nM T83011 CAY8X2 136032527 IC50 = 52480.75 nM T83011 C7YBC9 136032563 IC50 = 831.76 nM T83011 CX0Y7D 136032606 IC50 = 269.15 nM T83011 CRI68P 136035753 IC50 = 1283 nM T83011 C56NWE 136035754 IC50 = 369 nM T83011 C94ZQS 136035755 IC50 = 81 nM T83011 CFAB82 136035756 IC50 = 841 nM T83011 C2L8UX 136074346 Ki = 1640000 nM T83011 C8E2KH 136074347 Ki = 1480 nM T83011 CX95EP 136092233 IC50 = 83000 nM T83011 CA3JC8 136118613 IC50 = 37000 nM T83011 CQ2GP6 136118614 IC50 = 4300 nM T83011 C6R4IC 136118615 IC50 = 14267 nM T83011 CS0JL5 136118616 IC50 = 26333 nM T83011 C8RH6M 136118617 IC50 = 11633 nM T83011 CN4U6K 136118618 IC50 = 2667 nM T83011 CHWC38 136118619 IC50 = 12833 nM T83011 C5UDW3 136118620 IC50 = 51167 nM T83011 C8I6UN 136118621 IC50 = 3117 nM T83011 CV4E6W 136118635 IC50 = 450 nM T83011 CFI2X7 136118636 IC50 = 2567 nM T83011 CYS3M8 136118637 IC50 = 1237 nM T83011 C0UH1B 136118638 IC50 = 3733 nM T83011 C6G4AY 136118639 IC50 = 8750 nM T83011 C40VES 136118640 IC50 = 1417 nM T83011 CH4Q8O 136118646 IC50 = 2433 nM T83011 C43JTG 136118647 IC50 = 6000 nM T83011 CLH0V9 136118648 IC50 = 7033 nM T83011 C76XEJ 136118649 IC50 = 2000 nM T83011 CN0V5C 136118650 IC50 = 20700 nM T83011 CR72MQ 136118651 IC50 = 26000 nM T83011 CD7OE2 136118652 IC50 = 26833 nM T83011 CG5TX8 136118653 IC50 = 16767 nM T83011 CCHM67 136118657 IC50 = 4260 nM T83011 C0W1TM 136118658 IC50 = 5217 nM T83011 C40LYH 136118659 IC50 = 370 nM T83011 CZ7C3Y 136118660 IC50 = 207 nM T83011 C42FCS 136118661 IC50 = 2817 nM T83011 CR3DK1 136118716 IC50 = 28333 nM T83011 CON04G 136118728 IC50 = 25333 nM T83011 COX1F8 136118729 IC50 = 27800 nM T83011 CY5GU4 136118730 IC50 > 100000 nM T83011 C0R5PV 136118732 IC50 = 34333 nM T83011 CLU47S 136203753 IC50 = 173.78 nM T83011 CG9QT7 136203754 IC50 = 8709.64 nM T83011 C2UJA5 136203790 IC50 = 60255.96 nM T83011 C5SH0A 136219375 Ki = 6000 nM T83011 C4RP7K 136219376 Ki = 530000 nM T83011 CU7FD9 136232997 IC50 = 26800 nM T83011 CWE0G8 136232998 IC50 = 3040 nM T83011 CXG9N1 136232999 IC50 = 3170 nM T83011 CMPU87 136233000 IC50 = 3650 nM T83011 C3AIC2 136233006 IC50 = 5780 nM T83011 C7MLI3 136233007 IC50 = 1910 nM T83011 CK68XF 136233008 IC50 = 10440 nM T83011 CS81JR 136233009 IC50 = 2070 nM T83011 CE76VG 136233010 IC50 = 2640 nM T83011 CRPG40 136233012 IC50 = 3870 nM T83011 C8KWN7 136233016 IC50 = 20080 nM T83011 CNGU52 136233017 IC50 = 490 nM T83011 CQK12T 136233018 IC50 = 2040 nM T83011 C9LR0M 136233021 IC50 = 300 nM T83011 C20ULD 136233022 IC50 = 180 nM T83011 CI1XO6 136233023 IC50 = 340 nM T83011 CPZ80S 136239406 Ki = 305000 nM T83011 CEPX06 136239508 Ki = 11000 nM T83011 C5W8GX 136242978 Ki = 45000 nM T83011 CT7LY9 136242979 Ki = 56000 nM T83011 C6K3SZ 136244520 Ki = 15550 nM T83011 CA91YM 136260057 IC50 = 1882 nM T83011 C8D6CP 136260064 IC50 = 571 nM T83011 C8XZR1 136260489 Ki = 5000 nM T83011 CXM62D 136270607 Ki = 33500 nM T83011 CFP60G 136607463 IC50 = 168000 nM T83011 C6UID3 136686111 IC50 = 5990 nM T83011 CQ29VE 136966266 IC50 = 217 nM T83011 CDQ9R2 136966267 IC50 = 3422 nM T83011 CDFQ92 136966268 IC50 = 481 nM T83011 CHJI26 136966269 IC50 = 118 nM T83011 C30VEZ 136966270 IC50 = 388 nM T83011 CXY7K9 136966271 IC50 = 512 nM T83011 CHP3N6 136986940 Ki = 5230 nM T83011 C0ORN6 136986942 Ki = 990 nM T83011 C0GT6R 136986944 Ki = 750 nM T83011 CD1EU8 136986946 Ki = 20000 nM T83011 CX4CS1 136986948 Ki = 72000 nM T83011 C5GHZ1 136986950 Ki = 2000 nM T83011 CU2T7W 136986952 Ki = 14000 nM T83011 CVA2W6 136986954 Ki = 60000 nM T83011 C1HI9Q 136986956 Ki = 29660 nM T83011 C6TYF4 137174990 Ki = 350 nM T83011 C4ZKC3 137175204 Ki = 41050 nM T83011 C5A8RL 137175205 Ki = 15900 nM T83011 C1PE4I 137175206 Ki = 5900000 nM T83011 CKS92O 137175207 Ki = 4000 nM T83011 C36LNB 137175235 Ki = 201250 nM T83011 C2FMA0 137175236 Ki = 27950 nM T83011 C7YZF2 137175237 Ki = 2780 nM T83011 CVP1K0 137175238 Ki = 201350 nM T83011 C9P4YE 137459864 IC50 > 31622.78 nM T83011 CC5XJ7 137629431 IC50 = 24050 nM T83011 CIP6T2 137631403 IC50 = 262 nM T83011 CLVQ93 137631579 IC50 = 554 nM T83011 CE6L8G 137631680 IC50 = 18489 nM T83011 C74HIO 137631707 IC50 = 825 nM T83011 CW0BZ8 137631800 IC50 = 192 nM T83011 C9BXC6 137632300 IC50 = 590 nM T83011 CELH07 137632760 IC50 = 39 nM T83011 C5RC7Q 137633047 IC50 = 16700 nM T83011 C7TB1N 137633079 IC50 = 75 nM T83011 CP43GR 137633264 IC50 = 7300 nM T83011 CZ2HK3 137633315 IC50 = 2033 nM T83011 CM79NG 137633355 IC50 = 30800 nM T83011 CSY95X 137633406 IC50 = 12000 nM T83011 CDA65L 137633416 IC50 > 10000 nM T83011 C1D9FT 137633537 IC50 = 8100 nM T83011 CEI0T6 137633782 IC50 = 4700 nM T83011 CPEG26 137633844 IC50 = 18 nM T83011 C9RF5Z 137633956 IC50 = 6900 nM T83011 C6XUF8 137633971 IC50 = 390 nM T83011 C7WEV4 137634210 IC50 = 7600 nM T83011 C0C6NP 137634473 IC50 >= 1000000 nM T83011 CXA2E5 137634675 IC50 = 7600 nM T83011 CM2CR5 137635058 IC50 = 13450 nM T83011 C8IZ6F 137635535 IC50 = 6090 nM T83011 C20CWR 137635957 IC50 = 14300 nM T83011 CBQ27R 137636063 IC50 = 1880 nM T83011 CF6ZK2 137636117 IC50 = 13 nM T83011 CWLK63 137636137 Ki = 2.69 nM T83011 C4LS1I 137636518 IC50 = 380 nM T83011 C31QAB 137636695 IC50 = 4300 nM T83011 CB08HD 137636701 IC50 = 19200 nM T83011 CUR9N8 137636817 IC50 = 11300 nM T83011 CU4A5C 137636900 IC50 >= 1000000 nM T83011 COZ4G1 137636952 IC50 = 24900 nM T83011 CU5T9E 137636999 IC50 = 392 nM T83011 CXDG98 137637036 IC50 = 6500 nM T83011 CM35CX 137637171 IC50 = 1270 nM T83011 C9KOA0 137637296 IC50 = 173 nM T83011 C0N3UQ 137637571 IC50 = 21400 nM T83011 CNEH91 137637802 IC50 = 18600 nM T83011 CIH2B0 137637832 IC50 = 25 nM T83011 CBMA21 137638039 IC50 = 41.8 nM T83011 C39LZK 137638049 IC50 = 13100 nM T83011 CBZ3T5 137638261 IC50 = 106 nM T83011 C4HWF2 137638562 IC50 = 15100 nM T83011 CC85LZ 137638918 IC50 = 287 nM T83011 CQ8IR3 137638955 IC50 = 4 nM T83011 C4AX5H 137639047 IC50 = 9400 nM T83011 C9CYA8 137639104 IC50 = 2690 nM T83011 CY6VP5 137639127 IC50 > 25000 nM T83011 C3XTD6 137639448 IC50 = 21.8 nM T83011 C70NHU 137639458 IC50 = 350 nM T83011 C1A8CF 137639477 IC50 = 12200 nM T83011 C3XP6B 137639555 IC50 = 10151 nM T83011 C20ZJX 137640020 IC50 = 11300 nM T83011 C29UYV 137640667 IC50 = 634 nM T83011 CVF68A 137640689 IC50 = 4360 nM T83011 C5ZV1Y 137640778 IC50 = 3550 nM T83011 CV20WQ 137641088 IC50 = 9100 nM T83011 C06FVA 137641098 IC50 = 45.4 nM T83011 C0P7HY 137641250 IC50 = 3.94 nM T83011 C0CDW6 137641345 IC50 = 6500 nM T83011 CRS6D9 137641513 IC50 = 3730 nM T83011 C0TO4M 137641830 IC50 = 15900 nM T83011 CXK9D2 137641978 IC50 = 113.5 nM T83011 CSZ3O5 137642116 IC50 = 78.22 nM T83011 C8GYQ2 137642138 IC50 = 551 nM T83011 COX50U 137642409 IC50 = 330 nM T83011 CY70KG 137642691 IC50 = 20700 nM T83011 C7P6FH 137642777 IC50 = 12162 nM T83011 COW6Y8 137643059 IC50 > 10000 nM T83011 C68RZL 137643060 IC50 = 288 nM T83011 CL7K3X 137643291 IC50 = 73 nM T83011 CR4PY5 137643351 IC50 = 1780 nM T83011 C1E9CL 137644000 IC50 = 4000 nM T83011 C4AGP8 137644230 IC50 = 2340 nM T83011 CQCJ76 137644241 IC50 = 26800 nM T83011 CC03ZF 137644660 IC50 = 338 nM T83011 C0O2BL 137644693 IC50 = 12 nM T83011 C7TWP1 137644997 IC50 = 11700 nM T83011 CI2X8P 137645001 IC50 = 5600 nM T83011 C8W7CD 137645972 IC50 = 8200 nM T83011 CAC64D 137645994 IC50 = 8120 nM T83011 CYK7D5 137646140 IC50 = 8900 nM T83011 CUG5D3 137646552 IC50 = 6100 nM T83011 C0P8ED 137646555 IC50 = 8300 nM T83011 CR60SF 137646770 IC50 = 1700 nM T83011 CMX01E 137646776 IC50 = 26100 nM T83011 CG1P3T 137646871 IC50 = 165 nM T83011 CL3GO5 137647142 IC50 = 45.42 nM T83011 C0OEH1 137647178 IC50 = 1780 nM T83011 C97WYL 137647179 IC50 = 542 nM T83011 C4A6GE 137647180 IC50 > 10000 nM T83011 CTA0J8 137647190 IC50 = 2.2 nM T83011 C1D8NJ 137647314 IC50 = 12615 nM T83011 C5RLG0 137647656 IC50 = 881 nM T83011 C23JNQ 137647691 IC50 = 15500 nM T83011 C0YN6K 137647773 IC50 = 2500 nM T83011 CBR72P 137648289 IC50 = 12600 nM T83011 CD6T4U 137648513 IC50 = 15200 nM T83011 C4VQK8 137648638 IC50 = 2020 nM T83011 CSO5A1 137648685 IC50 = 2920 nM T83011 CUV07X 137649344 IC50 = 34600 nM T83011 C3WG5E 137649658 IC50 = 10333 nM T83011 CO3E6R 137649886 IC50 = 9400 nM T83011 C03HQU 137649999 IC50 = 1290 nM T83011 C4N1CL 137650217 IC50 = 5900 nM T83011 CG4XY5 137650246 IC50 = 764 nM T83011 CR61GZ 137650279 IC50 = 460 nM T83011 C0S8OQ 137650303 IC50 = 565 nM T83011 CZ96CG 137650801 IC50 = 8500 nM T83011 CJW29P 137650881 IC50 = 2600 nM T83011 C4OGA9 137651393 IC50 = 210.8 nM T83011 CSD27L 137651785 IC50 = 4228 nM T83011 C5LMU7 137651876 IC50 = 1120 nM T83011 C4UG6F 137651890 IC50 > 100000 nM T83011 CFXL04 137652113 IC50 = 1967 nM T83011 CH5EM3 137652372 IC50 = 10.31 nM T83011 CQ9B8K 137652578 IC50 = 370 nM T83011 CQ84TK 137652979 IC50 = 2891 nM T83011 C4AET5 137653036 IC50 = 25235 nM T83011 C7ANF0 137653292 IC50 = 3500 nM T83011 CLO76S 137653476 IC50 = 11700 nM T83011 C6R2QD 137653751 IC50 = 2200 nM T83011 C9NKO3 137653809 IC50 = 273 nM T83011 CES62O 137653949 IC50 = 1945 nM T83011 CS46QP 137654687 IC50 = 2030 nM T83011 CG0YV5 137655066 IC50 = 19200 nM T83011 C8AT6V 137655437 IC50 = 17.1 nM T83011 C38WAR 137655553 IC50 = 7130 nM T83011 CA1K3D 137655576 IC50 = 8600 nM T83011 C6RN4D 137655667 IC50 = 103 nM T83011 C9Q4BS 137655777 IC50 = 1526 nM T83011 C0R6HE 137655915 IC50 = 270 nM T83011 CQ0EP9 137656002 IC50 = 512.6 nM T83011 C0F7BV 137656084 IC50 = 6800 nM T83011 CTM8B1 137656100 IC50 = 5330 nM T83011 CUZJ29 137656171 IC50 = 1640 nM T83011 CK93UH 137656494 IC50 = 21500 nM T83011 C4F2WI 137656817 IC50 = 22 nM T83011 CJL6G1 137657126 IC50 = 14500 nM T83011 C46JPC 137657652 IC50 = 6300 nM T83011 C79ECM 137657666 IC50 = 3280 nM T83011 C81NJW 137657973 IC50 = 17000 nM T83011 C0VPL8 137658080 IC50 = 257 nM T83011 CB6DH1 137658226 IC50 = 5240 nM T83011 CI8W0P 137658678 IC50 = 2800 nM T83011 CQ1G8S 137658745 IC50 = 10100 nM T83011 CUT45L 137658804 IC50 = 18300 nM T83011 CZP1H6 137658871 IC50 = 7590 nM T83011 C6XDF0 137658917 IC50 >= 1000000 nM T83011 C0X6QO 137659176 IC50 = 31700 nM T83011 CFD5A3 137659177 IC50 >= 100000 nM T83011 CZL1Y8 137659445 IC50 = 3692 nM T83011 C7UHX3 137659615 IC50 = 880 nM T83011 C4NAO0 137659819 IC50 = 6420 nM T83011 CBD24K 137660365 IC50 = 12200 nM T83011 CG3M6F 137660472 IC50 = 915 nM T83011 CE0VO7 137660963 IC50 = 1130 nM T83011 CS2W1X 137661035 IC50 = 1730 nM T83011 CSM2V9 137661192 IC50 = 12860 nM T83011 C9VSC4 137661292 IC50 = 2270 nM T83011 C57MXQ 137661372 IC50 = 433 nM T83011 CU4Y6A 137661395 IC50 = 26600 nM T83011 CSU21O 137661504 IC50 = 3800 nM T83011 CAWM79 137661642 IC50 = 9100 nM T83011 CY94MB 137661806 IC50 = 6100 nM T83011 CJS6U1 137662125 IC50 = 284 nM T83011 C5OWM7 137662199 IC50 = 674.2 nM T83011 C1W7ZD 137662235 IC50 = 621.7 nM T83011 C16IHB 137662240 IC50 = 136 nM T83011 C04JHX 139087190 IC50 = 7.3 nM T83011 C35ARK 139087191 IC50 = 1.148 nM T83011 C3AB1I 139087386 IC50 = 1.318 nM T83011 CQ5W3D 139449915 IC50 = 136 nM T83011 CMG0D5 141488053 IC50 = 4570 nM T83011 CIN08E 141520106 IC50 = 21100 nM T83011 CR8W6O 141520108 IC50 = 3660 nM T83011 CN1TV3 141520110 IC50 = 35980 nM T83011 CFYM37 141520115 IC50 = 4620 nM T83011 C0R3XT 141520119 IC50 = 94020 nM T83011 C02TUS 141520121 IC50 = 151100 nM T83011 CE3FU5 141520123 IC50 = 14080 nM T83011 CKS8R1 141520127 IC50 = 71380 nM T83011 CX3DI7 141520133 IC50 > 200000 nM T83011 CUZ2C8 141766036 IC50 = 240 nM T83011 CA7H1W 141766041 IC50 = 180 nM T83011 CC0YW1 145946358 IC50 > 1000 nM T83011 CQBR80 145946627 IC50 > 1000 nM T83011 C1LZ8S 145946736 IC50 > 1000 nM T83011 CH86KT 145946845 IC50 = 1228 nM T83011 C5NAF3 145946984 IC50 > 1000 nM T83011 CAO76Z 145947001 IC50 = 1495 nM T83011 C1BUS5 145947244 IC50 > 1000 nM T83011 CKE7X5 145947256 IC50 > 1000 nM T83011 C4TM6G 145947709 IC50 > 1000 nM T83011 CXF8J0 145947753 IC50 > 1000 nM T83011 C3RP4B 145947772 IC50 > 1000 nM T83011 C7GI9D 145947814 IC50 = 609 nM T83011 C48YVA 145947815 IC50 = 1128 nM T83011 CXZV16 145947948 IC50 > 1000 nM T83011 C95DIF 145947967 IC50 > 1000 nM T83011 C62TCL 145947968 IC50 > 1000 nM T83011 C02PUB 145948036 IC50 > 1000 nM T83011 C1AXM6 145948069 IC50 = 390 nM T83011 CY3A7G 145948500 IC50 = 5.5 nM T83011 CKT3V1 145948504 IC50 = 4200 nM T83011 CT48HM 145948506 IC50 = 400 nM T83011 C4C1JY 145948507 IC50 = 620 nM T83011 CM7FE5 145948508 IC50 = 1400 nM T83011 CJ4Q9L 145948509 IC50 = 850 nM T83011 CHFL20 145948511 IC50 = 2100 nM T83011 CEIL06 145948520 IC50 = 350 nM T83011 CQOP12 145948521 IC50 = 440 nM T83011 C71JXN 145948522 IC50 = 250 nM T83011 C8I4CY 145948524 IC50 = 39 nM T83011 C4C7VQ 145948525 IC50 = 130 nM T83011 CSR05F 145948530 IC50 = 91 nM T83011 CZJ2M5 145948531 IC50 = 3100 nM T83011 C13EJK 145948532 IC50 = 61 nM T83011 CC2N4S 145948533 IC50 = 230 nM T83011 COL6M1 145948534 IC50 = 100 nM T83011 CJD26S 145948549 IC50 = 83 nM T83011 CZ61JB 145948550 IC50 = 120 nM T83011 C81KYR 145948553 IC50 = 26 nM T83011 CVF2R3 145948554 IC50 = 1200 nM T83011 CD83FI 145948555 IC50 = 160 nM T83011 C7ID5T 145948556 IC50 = 200 nM T83011 CJ8PF4 145948559 IC50 = 63 nM T83011 C7IX0H 145948560 IC50 = 590 nM T83011 CK21IG 145948561 IC50 = 2500 nM T83011 CW3CF1 145948562 IC50 = 71 nM T83011 C97JVF 145948622 IC50 = 30000 nM T83011 C9XO4M 145948655 IC50 = 29000 nM T83011 CHP2V5 145948690 IC50 > 30000 nM T83011 CLD12N 145949023 IC50 = 30000 nM T83011 C5GM0U 145949030 IC50 > 30000 nM T83011 C1TDL9 145949549 IC50 = 5.3 nM T83011 CDA28I 145949712 IC50 = 87090 nM T83011 CM12NP 145949823 IC50 > 1000000 nM T83011 C54UIF 145949921 IC50 = 182 nM T83011 CRN6H7 145949934 IC50 = 5520 nM T83011 CPX50L 145949947 IC50 > 50000 nM T83011 CW3P6G 145950085 IC50 = 550 nM T83011 CGQ3U6 145950141 IC50 = 3870 nM T83011 C81JWA 145950243 IC50 > 50000 nM T83011 CO2M5E 145950303 IC50 > 100000 nM T83011 C49AIV 145950338 IC50 = 12 nM T83011 CRD3S7 145950766 IC50 = 2990 nM T83011 CC7Q3F 145950843 IC50 = 12435 nM T83011 C8SM2O 145950855 IC50 = 6110 nM T83011 CX91AI 145950913 IC50 = 2490 nM T83011 C1VE0Q 145951053 IC50 = 6990 nM T83011 C8RQ2P 145951193 IC50 = 14574 nM T83011 CM3R8C 145951251 IC50 > 50000 nM T83011 C3U0WI 145951283 IC50 = 3270 nM T83011 CJN6H5 145951347 IC50 = 1090 nM T83011 CY91WG 145951519 IC50 > 50000 nM T83011 CAY7P0 145951540 IC50 > 50000 nM T83011 CO4X0H 145951870 IC50 = 2510 nM T83011 CX1P7H 145952331 IC50 > 100000 nM T83011 C8YD1P 145952456 IC50 = 5380 nM T83011 C19ZGF 145952532 IC50 = 5236 nM T83011 C47ABX 145952713 IC50 = 7.2 nM T83011 CA0H2O 145952896 IC50 > 1000000 nM T83011 C8LU9S 145953219 IC50 = 557921 nM T83011 CFE03V 145953575 IC50 = 6240 nM T83011 CCG6Z2 145953702 IC50 > 50000 nM T83011 CN47FR 145953732 IC50 = 4340 nM T83011 CJ1XM7 145953859 IC50 = 4150 nM T83011 CM3T6Y 145953870 IC50 = 750 nM T83011 CRYS31 145954037 IC50 = 1760 nM T83011 CCV17M 145954104 IC50 = 3830 nM T83011 C1I9WM 145954115 IC50 = 1970 nM T83011 CUMJ40 145954156 IC50 = 130675 nM T83011 CL0XT8 145954248 IC50 > 100000 nM T83011 CC9A0N 145954291 IC50 = 110 nM T83011 CUIY71 145954565 IC50 > 50000 nM T83011 CZ5MI9 145954575 IC50 = 1427 nM T83011 C3FS2N 145954793 IC50 = 770 nM T83011 C8A4TF 145954923 IC50 = 6910 nM T83011 CVBH34 145954971 IC50 > 50000 nM T83011 C90TGE 145955059 IC50 = 6910 nM T83011 C8FSO7 145955146 IC50 = 6210 nM T83011 CE8G4I 145955186 IC50 > 100000 nM T83011 CZU84I 145955291 IC50 > 1000000 nM T83011 CKU7Z5 145955423 IC50 = 355 nM T83011 C37SYH 145955424 IC50 > 100000 nM T83011 CCZ2R9 145955785 IC50 = 3130 nM T83011 CRTP17 145955809 IC50 = 10220 nM T83011 C2DF7C 145955811 IC50 = 1410 nM T83011 CQ6MY0 145956006 IC50 = 17615 nM T83011 C5XT4Z 145956132 IC50 > 100000 nM T83011 CHEG86 145956238 IC50 = 118 nM T83011 CPY71F 145956290 IC50 > 100000 nM T83011 C4MUO0 145956291 IC50 = 6210 nM T83011 C2XOL5 145956393 IC50 > 50000 nM T83011 CDY0S5 145956567 IC50 = 1680 nM T83011 C28IPH 145957131 IC50 = 2890 nM T83011 C0U5NS 145957329 IC50 = 20900 nM T83011 C9W6MV 145957333 IC50 = 8.6 nM T83011 CGO4F6 145957401 IC50 = 640 nM T83011 CJ03TU 145957740 IC50 > 100000 nM T83011 C9ES7D 145957769 IC50 = 760721 nM T83011 C4G3LT 145957957 IC50 = 10490 nM T83011 CN4R9J 145958017 IC50 = 5870 nM T83011 CY4EX0 145958214 IC50 = 330 nM T83011 CUJQ65 145958271 IC50 = 10 nM T83011 CC18RP 145958787 IC50 > 50000 nM T83011 CGD7Z3 145958889 IC50 = 430 nM T83011 C93IGN 145958945 IC50 = 650 nM T83011 C25OZA 145958966 IC50 = 141041 nM T83011 C5A1TY 145959187 IC50 = 1390 nM T83011 CZ1O7J 145959317 IC50 = 3229 nM T83011 C0M7PW 145959369 IC50 > 50000 nM T83011 CPF6B7 145959387 IC50 = 2910 nM T83011 C7DZA2 145959459 IC50 = 53 nM T83011 C9FQH0 145959513 IC50 = 1870 nM T83011 CV8Z4N 145959672 IC50 = 29500 nM T83011 CUXZ08 145959682 IC50 > 1000000 nM T83011 CB6O5R 145959714 IC50 = 55 nM T83011 C69BEI 145959843 IC50 = 133362 nM T83011 CYP62M 145959951 IC50 = 4720 nM T83011 CU58SO 145960091 IC50 = 3390 nM T83011 C37OHE 145960135 IC50 = 680 nM T83011 CL0WE8 145960174 IC50 = 101 nM T83011 C13WSY 145960214 IC50 = 626 nM T83011 CG5KQ7 145960277 IC50 > 50000 nM T83011 C4V1GR 145960343 IC50 = 47 nM T83011 C62JCL 145960933 IC50 = 410 nM T83011 C59ASP 145961050 IC50 > 10000 nM T83011 C2BZ5C 145961747 IC50 > 10000 nM T83011 CTRZ67 145961995 IC50 = 7000 nM T83011 CFM39D 145962916 IC50 = 2390 nM T83011 CLB9Q2 145962957 IC50 > 10000 nM T83011 CU12MA 145963481 IC50 > 10000 nM T83011 CD39PS 145963747 IC50 = 280 nM T83011 CTH70Y 145963788 IC50 = 3990 nM T83011 C25IUB 145963838 IC50 = 13540 nM T83011 CQ5RX2 145964047 IC50 = 1507 nM T83011 C8E3AJ 145964075 IC50 = 17000 nM T83011 C9RC3Y 145964200 IC50 = 3880 nM T83011 CF6Q8B 145964244 IC50 = 7381 nM T83011 C4KW1B 145964292 IC50 = 31000 nM T83011 CD2X4I 145964386 IC50 = 37000 nM T83011 CH5G8U 145964572 IC50 = 978 nM T83011 CG5FA8 145964757 IC50 = 3160 nM T83011 C7KMT6 145964810 IC50 = 15460 nM T83011 CXJS15 145964929 IC50 > 10000 nM T83011 CZE6R5 145965009 IC50 = 175 nM T83011 C9V4IH 145965010 IC50 = 5643 nM T83011 C2CL8F 145965108 IC50 = 6078 nM T83011 C7T5SN 145965193 IC50 = 24430 nM T83011 C7GF1E 145965278 IC50 = 1131 nM T83011 CLW9H6 145965317 IC50 = 5530 nM T83011 CVYM98 145965396 IC50 = 5757 nM T83011 CMED83 145965605 IC50 = 3900 nM T83011 CMYG28 145965829 IC50 = 5003 nM T83011 CTS35V 145966018 IC50 = 1803 nM T83011 CP2S1C 145966310 IC50 = 24800 nM T83011 CF06BV 145966566 IC50 = 58000 nM T83011 C4W0RU 145966651 IC50 = 8800 nM T83011 CAX84N 145966790 IC50 = 283 nM T83011 CS5FC0 145966840 IC50 = 2110 nM T83011 C5D3HZ 145966917 IC50 > 10000 nM T83011 CB71YE 145966926 IC50 = 4855 nM T83011 C9QJL3 145967042 IC50 = 2160 nM T83011 CZES12 145967115 IC50 = 1085 nM T83011 C60ZBC 145967151 IC50 = 6958 nM T83011 C32VEK 145967213 IC50 = 23570 nM T83011 CIRD04 145967411 IC50 = 3146 nM T83011 CIXR60 145967524 IC50 = 396 nM T83011 CHTN65 145967763 IC50 = 11100 nM T83011 C03CRW 145968128 IC50 = 19200 nM T83011 CWJ64D 145968255 IC50 = 8600 nM T83011 CK5VJ2 145968464 IC50 = 19170 nM T83011 CWX75L 145968655 IC50 = 12400 nM T83011 CB80FD 145968869 IC50 = 18800 nM T83011 CQV1S7 145969296 IC50 > 100000 nM T83011 CR8Z2D 145969616 IC50 = 2190 nM T83011 CYMF27 145969637 IC50 = 1568 nM T83011 CSXF25 145969647 IC50 = 20100 nM T83011 CY32TF 145969707 IC50 = 19400 nM T83011 C6M2FZ 145970256 IC50 = 13200 nM T83011 C6A4SV 145970363 IC50 = 20100 nM T83011 C27EMD 145970504 IC50 = 193 nM T83011 C67OFB 145970725 IC50 = 19600 nM T83011 C6PYZ0 145970731 IC50 = 13700 nM T83011 CW60FG 145970775 IC50 = 4000 nM T83011 C9IW2K 145970779 IC50 = 60000 nM T83011 C97VSH 145971024 IC50 = 541 nM T83011 C23KUV 145971152 IC50 = 19700 nM T83011 C6N7JF 145971479 IC50 = 42908 nM T83011 CVTO93 145971704 IC50 = 20 nM T83011 C3Q1TN 145971772 IC50 = 18010 nM T83011 C01DYM 145971895 IC50 = 15300 nM T83011 COE8K3 145971958 IC50 = 189 nM T83011 CKY7V1 145971968 IC50 = 53074 nM T83011 CUTB21 145972060 IC50 = 8340 nM T83011 CQ7U1M 145972128 IC50 = 17000 nM T83011 C02NHL 145972143 IC50 = 2849 nM T83011 C19WJX 145972230 IC50 = 360 nM T83011 CPNJ15 145972300 IC50 = 110 nM T83011 CXIM57 145972351 IC50 = 1676 nM T83011 CO19QS 145972772 IC50 = 27 nM T83011 C4M1OA 145972797 IC50 = 560 nM T83011 CNE54W 145972804 IC50 > 10000 nM T83011 C6R8IL 145973192 IC50 = 425858 nM T83011 C5SM0J 145973231 IC50 = 6870 nM T83011 C9RFE4 145973241 IC50 = 2510 nM T83011 C1LM0W 145973337 IC50 = 7014 nM T83011 CP32EZ 145973435 IC50 = 2369 nM T83011 CJB7U5 145973747 IC50 = 6890 nM T83011 CNM9X5 145973760 IC50 = 10840 nM T83011 CE9JC0 145973764 IC50 = 3742 nM T83011 CAC9Q8 145973846 IC50 > 60000 nM T83011 CS41YW 145973896 IC50 = 3050 nM T83011 CB5H6K 145973982 IC50 = 4437 nM T83011 C6F1WT 145974014 IC50 = 3324 nM T83011 C1I3SB 145974077 IC50 > 100000 nM T83011 CYSL73 145974355 IC50 = 300 nM T83011 CY1G2F 145974565 IC50 > 100000 nM T83011 C1TI6B 145974586 IC50 > 10000 nM T83011 CFN8D6 145974596 IC50 > 100000 nM T83011 C8W2KY 145974736 IC50 = 37000 nM T83011 C08TXO 145974839 IC50 = 24620 nM T83011 C9EFC7 145974855 IC50 = 387 nM T83011 CGAP39 145974892 Ki = 2927 nM T83011 C1YRD3 145974906 IC50 = 3513 nM T83011 CU15SA 145974947 IC50 = 232 nM T83011 C7O4SQ 145974973 IC50 = 10000 nM T83011 CPD90H 145975028 IC50 = 17620 nM T83011 C3HPU6 145975029 IC50 = 3200 nM T83011 CTMD94 145975130 IC50 = 2890 nM T83011 CHZS47 145975154 IC50 = 4210 nM T83011 C4ZR8Y 145975227 IC50 = 1730 nM T83011 CO0D6E 145975284 IC50 = 1103 nM T83011 CR21PI 145975443 IC50 = 41 nM T83011 C7NV3M 145975746 IC50 = 4594 nM T83011 C7CW4G 145975882 IC50 = 8298 nM T83011 CZO18H 145976060 IC50 = 7580 nM T83011 C8JVC1 145976117 IC50 = 1570 nM T83011 CR2MT1 145976177 IC50 > 10000 nM T83011 CZYI64 145976195 IC50 = 1552 nM T83011 CCG38X 145976354 IC50 = 9625 nM T83011 C0AV1B 145976627 IC50 = 12850 nM T83011 CF6Y0W 145977123 IC50 = 22710 nM T83011 CI1WB7 145977381 IC50 = 13500 nM T83011 C59KDE 145977426 IC50 = 10140 nM T83011 CDH04P 145977491 IC50 = 1230 nM T83011 C8IAL2 145977624 IC50 = 262 nM T83011 CB53MH 145977978 IC50 = 2339 nM T83011 CV2TD0 145978096 IC50 = 2870 nM T83011 C9H1EZ 145978133 IC50 = 3495 nM T83011 C68MBY 145978156 IC50 = 6780 nM T83011 C93MSO 145978282 IC50 = 402 nM T83011 CX2O5U 145978432 IC50 = 2640 nM T83011 CZ7RE2 145978507 IC50 = 19150 nM T83011 CB4RK0 145978554 IC50 = 4000 nM T83011 C3WM4R 145978572 IC50 = 5350 nM T83011 CJ6TL1 145978580 IC50 = 30110 nM T83011 C1QE8L 145978587 IC50 > 10000 nM T83011 CST06V 145978709 IC50 = 750 nM T83011 CQZ0G5 145978902 IC50 = 13900 nM T83011 CHX28E 145978908 IC50 = 824 nM T83011 CHWP93 145979173 Ki = 6000000 nM T83011 CQG60B 145979201 IC50 > 100000 nM T83011 CJS5N8 145979426 IC50 > 100000 nM T83011 C4TR1C 145979433 IC50 = 2620 nM T83011 CQ30IN 145979533 Ki = 5771000 nM T83011 C7HTX2 145979575 IC50 = 56200 nM T83011 CH13FK 145979661 IC50 = 3680 nM T83011 C15CDR 145979739 IC50 = 200 nM T83011 C5BLA7 145979756 IC50 = 3650 nM T83011 CX2RW9 145979866 IC50 = 92100 nM T83011 C1D9ZU 145979972 IC50 = 56400 nM T83011 CLMR68 145980013 IC50 = 97500 nM T83011 CHRW12 145980490 IC50 = 85100 nM T83011 C0VAL8 145980562 IC50 = 9680 nM T83011 CW93VH 145980588 IC50 = 37900 nM T83011 CU0TA8 145980601 IC50 = 9300 nM T83011 CUI5C2 145980623 IC50 = 1400 nM T83011 C8D1JR 145981161 IC50 = 8610 nM T83011 CZ5H3I 145981171 IC50 = 89100 nM T83011 C87KIE 145981180 IC50 = 16520 nM T83011 CB9Q6H 145981331 IC50 = 8700 nM T83011 CN1RQ3 145981915 IC50 = 33500 nM T83011 CEM93S 145981925 IC50 = 89200 nM T83011 CX3M9J 145981988 IC50 = 571 nM T83011 CG1BW6 145982188 IC50 = 166 nM T83011 CS50XZ 145982212 IC50 = 13200 nM T83011 CZY08I 145982378 IC50 > 100000 nM T83011 CWNB08 145982383 IC50 = 2900 nM T83011 CFNJ87 145982457 IC50 > 100000 nM T83011 CAC72J 145982690 IC50 = 7200 nM T83011 CG34HN 145983490 IC50 > 200000 nM T83011 C7VJ1L 145983695 IC50 = 38.1 nM T83011 CO57QR 145984876 IC50 = 756 nM T83011 CAJ4D1 145986300 IC50 > 100000 nM T83011 CV46GJ 145986363 Ki = 140100 nM T83011 CCWA30 145986676 IC50 > 100000 nM T83011 CW3RG1 145987055 IC50 = 14100 nM T83011 C5A1VF 145987332 Ki = 4770160 nM T83011 CYWE49 145987379 IC50 = 12500 nM T83011 C21BYI 145987407 IC50 > 100000 nM T83011 CVM40C 145987439 IC50 = 9800 nM T83011 CX3CK0 145987477 IC50 = 880 nM T83011 CKV9T1 145987752 IC50 = 70400 nM T83011 C98DHT 145987800 IC50 = 71600 nM T83011 CA82TF 145987838 IC50 > 100000 nM T83011 C3M1ZO 145988042 IC50 = 51200 nM T83011 CVD20U 145988532 Ki = 478 nM T83011 CJ3L5S 145988539 IC50 = 22700 nM T83011 CNV67D 145988788 IC50 = 2210 nM T83011 C1XU7P 145988798 IC50 > 100000 nM T83011 CFQ97B 145989140 IC50 = 11700 nM T83011 CWJ1R2 145989205 IC50 = 7400 nM T83011 C2A8MY 145989254 IC50 = 48.4 nM T83011 C6L7UW 145989358 IC50 = 208 nM T83011 CUJ53A 145989396 IC50 = 10500 nM T83011 C4C2IS 145989399 IC50 = 12500 nM T83011 C6QRA9 145989946 IC50 = 2370 nM T83011 CTJ5L4 145989961 IC50 = 4660 nM T83011 C2AG8U 145990124 IC50 = 1250 nM T83011 CJFG45 145990271 IC50 = 95700 nM T83011 CSR71M 145990276 IC50 = 3220 nM T83011 CDIV28 145990279 IC50 = 46900 nM T83011 CR59TZ 145990611 IC50 > 100000 nM T83011 CQ4R9F 145990749 IC50 = 8500 nM T83011 CCAM14 145990761 IC50 = 4290 nM T83011 C5QZJ4 145990784 IC50 > 100000 nM T83011 CCMT53 145990789 IC50 = 43.8 nM T83011 CIFD61 145990950 IC50 = 1590 nM T83011 C10HQC 145991026 IC50 > 100000 nM T83011 CO5V7B 145991298 IC50 = 18200 nM T83011 CN9AG4 145991348 Ki = 68 nM T83011 C70GLU 145991351 IC50 = 1840 nM T83011 C3Y7FC 145991399 IC50 = 6700 nM T83011 CKQ9N2 145991501 IC50 = 2860 nM T83011 C1ZQ0W 145991508 IC50 = 2280 nM T83011 C1EH4M 145991565 IC50 = 6240 nM T83011 C9L8FJ 145991954 IC50 = 8900 nM T83011 CRWN45 145992049 IC50 = 3980 nM T83011 C1O3VK 145992136 IC50 = 37.2 nM T83011 CB9P8D 145992212 IC50 = 13600 nM T83011 CA75QO 145992385 IC50 = 700 nM T83011 CDI31H 145992535 IC50 = 38600 nM T83011 C1WI3A 145992723 IC50 = 5200 nM T83011 CJ04DE 145992806 IC50 = 11100 nM T83011 CUAI94 145992856 IC50 = 720 nM T83011 C1JW3O 145992909 IC50 = 250 nM T83011 CFE95O 145992966 IC50 > 100000 nM T83011 C4DBL8 145993064 IC50 = 43800 nM T83011 CIH8O3 145993065 IC50 = 3140 nM T83011 CV4AT0 145993142 Ki = 6000000 nM T83011 C5YMR4 145993208 IC50 > 100000 nM T83011 CY2N1D 145993326 Ki = 337 nM T83011 C18JHX 145993344 IC50 = 4520 nM T83011 CUVC73 145993378 IC50 > 100000 nM T83011 CVY1T9 145993407 IC50 = 28840 nM T83011 CLST75 145993460 IC50 = 950 nM T83011 C30CMY 145993498 IC50 > 100000 nM T83011 CYFO75 145993569 IC50 > 100000 nM T83011 C7H2UE 145993600 IC50 = 2540 nM T83011 CE0YD2 145993718 IC50 = 83400 nM T83011 C4HB6A 145993956 IC50 = 16400 nM T83011 CJZ10N 145994024 IC50 = 2280 nM T83011 CNY18A 145994134 IC50 = 3950 nM T83011 CRQ31D 145994230 IC50 = 2200 nM T83011 C4V2RJ 145994271 IC50 = 59900 nM T83011 CU9M1Y 145994293 IC50 = 6500 nM T83011 CXA07D 149927323 IC50 = 1745.3 nM T83011 C4NZ6L 150525142 IC50 > 50000 nM T83011 CI32AF 150615303 IC50 = 2280 nM T83011 CJE43S 150762943 IC50 = 30 nM T83011 CJR07T 150914951 IC50 = 230 nM T83011 C7E9LT 150956546 IC50 = 890 nM T83011 CSDW79 151032063 IC50 = 64 nM T83011 CP93LE 151074609 IC50 = 4280 nM T83011 CP8U5D 151566527 Ki = 38 nM T83011 C2U4KE 151661379 IC50 = 3640 nM T83011 CL2G3S 151810046 IC50 = 19162.8 nM T83011 CL8DP4 152061489 IC50 = 216 nM T83011 CZFU85 152109514 IC50 = 30 nM T83011 C7D4UB 152687816 IC50 > 50000 nM T83011 CP56CH 152688549 IC50 = 411 nM T83011 CJY38R 153525743 IC50 > 50000 nM T83011 C2FUG3 153525745 IC50 > 50000 nM T83011 CJM37F 153525746 IC50 > 50000 nM T83011 C5MCK8 153525747 IC50 > 50000 nM T83011 C2ZI9B 153525748 IC50 = 38900 nM T83011 C67IQJ 153525750 IC50 > 50000 nM T83011 CGP93O 153525752 IC50 > 50000 nM T83011 CS7F8Q 153525754 IC50 > 50000 nM T83011 C7U4GO 153525755 IC50 > 50000 nM T83011 CM97FW 153525756 IC50 > 50000 nM T83011 CQ4R8G 153525759 IC50 = 5500 nM T83011 CD81MP 153525760 IC50 > 50000 nM T83011 CS0ZN7 153525761 IC50 = 4100 nM T83011 CU16IY 153525763 IC50 > 50000 nM T83011 C6ZDG0 153525764 IC50 = 1000 nM T83011 C02PQN 153525765 IC50 > 50000 nM T83011 CFR4W2 153525769 IC50 > 50000 nM T83011 CIVC40 153525771 IC50 = 1000 nM T83011 CD0J3R 153525775 IC50 > 50000 nM T83011 C1NK6C 153525776 IC50 > 50000 nM T83011 CJ26VA 153525778 IC50 = 21000 nM T83011 CS6N2Z 153525780 IC50 > 50000 nM T83011 CCI3U5 153525781 IC50 = 16100 nM T83011 CBV4E7 153525782 IC50 > 50000 nM T83011 CMJQ60 153525784 IC50 > 50000 nM T83011 CM87OZ 153525785 IC50 > 50000 nM T83011 C6T9SI 153525786 IC50 > 50000 nM T83011 CVG27E 153525788 IC50 > 50000 nM T83011 C2YWN9 153525789 IC50 > 50000 nM T83011 CBC36V 153525792 IC50 > 50000 nM T83011 C8IW1V 153525795 IC50 > 50000 nM T83011 CFH9L5 153525796 IC50 > 50000 nM T83011 C4V7YJ 155510534 IC50 = 1600 nM T83011 C52SJA 155510567 IC50 > 100000 nM T83011 CV02GT 155510689 IC50 = 318 nM T83011 C9ATE6 155510755 IC50 = 6700 nM T83011 C0FHD2 155510783 IC50 = 14200 nM T83011 CB74UX 155510892 IC50 = 1490 nM T83011 CRI91T 155511196 IC50 = 20 nM T83011 CP5OS6 155511517 IC50 > 100000 nM T83011 C1NE6X 155511966 IC50 = 100000 nM T83011 C14FHM 155512092 IC50 > 50000 nM T83011 CI0DK6 155512416 IC50 = 11229.4 nM T83011 C54NIK 155512517 IC50 = 6050 nM T83011 C8Z1IA 155512624 IC50 = 730 nM T83011 CW6C3Q 155512810 IC50 > 100000 nM T83011 C9VTC4 155513287 IC50 = 13800 nM T83011 C21PXB 155513855 IC50 = 2.7 nM T83011 CDLC76 155513877 IC50 = 163 nM T83011 C9UT6Z 155513926 IC50 = 3930 nM T83011 CKVM85 155514248 IC50 > 10000 nM T83011 CTQ3F4 155514293 IC50 = 95610 nM T83011 C9X5TG 155514592 IC50 = 32.7 nM T83011 CRJ0A3 155514729 IC50 = 15800 nM T83011 C5AT7Z 155514789 IC50 > 20000 nM T83011 C3VYW4 155514859 IC50 = 14130 nM T83011 C3HE8N 155515066 IC50 = 274 nM T83011 C3I9WB 155515459 IC50 = 137 nM T83011 CR7C0G 155515606 IC50 = 53900 nM T83011 CYAI06 155515670 IC50 = 7100 nM T83011 CEBX27 155515845 IC50 = 120.9 nM T83011 C1F6GM 155515963 IC50 = 40250 nM T83011 CNV02U 155516016 IC50 = 385 nM T83011 C7BF6M 155516327 IC50 = 300 nM T83011 CJ1PQ3 155516433 IC50 = 18500 nM T83011 CO9PI2 155516509 IC50 > 10000 nM T83011 CPBN03 155516779 IC50 = 110 nM T83011 CAQ9G2 155516780 IC50 = 196 nM T83011 C5QJ4R 155516939 IC50 = 10000 nM T83011 CEA8D5 155516976 IC50 = 608 nM T83011 C0N9ZD 155517085 IC50 = 53000.5 nM T83011 CAH53U 155517120 IC50 > 10000 nM T83011 C4SK9Z 155517252 IC50 = 320 nM T83011 CTE5N3 155517491 IC50 = 34300 nM T83011 CUAG18 155517670 IC50 = 160 nM T83011 CNR5S8 155517867 IC50 = 128.6 nM T83011 C5PO3X 155517932 IC50 = 279000 nM T83011 C8JMD2 155518028 IC50 = 10200 nM T83011 C2CWD9 155518118 IC50 = 18070 nM T83011 CIM31H 155518405 IC50 = 10300 nM T83011 C0N3GJ 155518426 IC50 = 800 nM T83011 CKC0J2 155518449 IC50 = 66720 nM T83011 CHQX97 155518786 IC50 = 50 nM T83011 CGLO35 155518855 IC50 = 13800 nM T83011 C3SAR7 155519016 IC50 > 10000 nM T83011 CW7TP1 155519024 IC50 > 100000 nM T83011 C36LGV 155519027 IC50 = 28770 nM T83011 CR9ZW6 155519043 IC50 = 36 nM T83011 CIN90T 155519865 IC50 = 710 nM T83011 C5MV7W 155519920 IC50 = 1800 nM T83011 CP8UD6 155520012 IC50 = 21600 nM T83011 C3B0WM 155520213 IC50 = 1260 nM T83011 CM92LW 155520339 IC50 = 6300 nM T83011 C2GAV1 155520534 IC50 = 22 nM T83011 C76VBO 155520546 IC50 = 22120 nM T83011 CY25CV 155520663 IC50 > 10000 nM T83011 C7R8UB 155520744 IC50 > 10000 nM T83011 CRBE64 155520811 IC50 = 970 nM T83011 CLN8H5 155520953 IC50 = 76 nM T83011 CXW82M 155520967 IC50 = 3650 nM T83011 C3DZQ4 155521124 IC50 = 48912 nM T83011 CAC2H5 155521304 IC50 = 7590 nM T83011 CF28LO 155521322 IC50 = 21080 nM T83011 CP0E2K 155521356 IC50 = 76 nM T83011 C5ICT0 155521473 IC50 = 14900 nM T83011 C7M1BD 155521481 IC50 = 1100 nM T83011 C86WXD 155521569 IC50 = 297 nM T83011 CPM03G 155521729 Ki = 53.5 nM T83011 C2V8SU 155521773 IC50 > 10000 nM T83011 CEAV65 155521960 IC50 = 1370 nM T83011 C4YPF9 155522024 IC50 > 50000 nM T83011 CLK83G 155522136 IC50 = 7830 nM T83011 C3F1JX 155522174 IC50 = 9700 nM T83011 CCMY57 155522215 IC50 = 163.1 nM T83011 C4F7XP 155522484 IC50 = 250 nM T83011 CB57GS 155522741 IC50 = 48 nM T83011 C8ZOV5 155522894 IC50 = 36310 nM T83011 CTH80O 155523061 IC50 = 168 nM T83011 CB9F0K 155523307 IC50 = 223.1 nM T83011 CA4SQ3 155523568 IC50 = 1883.9 nM T83011 C93MOY 155523685 IC50 > 20000 nM T83011 C6U5XY 155523893 IC50 = 20030 nM T83011 C58KHY 155523916 IC50 = 4600 nM T83011 CKR9P2 155523992 IC50 = 660 nM T83011 C0JDC4 155524002 IC50 > 100000 nM T83011 CN3M7K 155524167 IC50 = 1500 nM T83011 C7STO9 155524244 IC50 = 876 nM T83011 CAT07S 155524254 IC50 = 2900 nM T83011 CED31W 155524277 IC50 = 34 nM T83011 CD3WT1 155524398 IC50 = 22090 nM T83011 CFJM83 155524430 IC50 = 980 nM T83011 CD24BF 155524446 IC50 = 2150 nM T83011 CRX87C 155524602 IC50 = 10970 nM T83011 CAEV51 155524611 IC50 = 1210 nM T83011 CI2U4J 155524971 IC50 = 29800 nM T83011 C1WZX5 155525062 IC50 = 10000 nM T83011 CS1LG9 155525089 IC50 = 41800 nM T83011 CKZD25 155525182 IC50 = 870 nM T83011 COKC12 155525316 IC50 = 5300 nM T83011 CI0V5F 155525579 IC50 > 100000 nM T83011 C4L0EO 155525604 IC50 = 13500 nM T83011 C9T3SC 155525695 IC50 = 14010 nM T83011 C2YS9O 155525759 IC50 = 30 nM T83011 C7IQ6J 155525760 IC50 = 23 nM T83011 CY0W2Z 155525787 IC50 > 10000 nM T83011 CT4XV9 155525799 IC50 = 12600 nM T83011 CQU8C1 155526013 IC50 = 7680 nM T83011 CNQ04W 155526184 IC50 = 74 nM T83011 CKA2M3 155526429 IC50 = 51 nM T83011 C9Q0OP 155526667 IC50 = 8090 nM T83011 CEBY20 155526946 IC50 = 22800 nM T83011 CY0P1G 155527083 IC50 = 132400 nM T83011 C2UO1C 155527178 IC50 = 190100 nM T83011 CLF6J9 155527441 IC50 = 210 nM T83011 C6J0FT 155527760 IC50 = 3300 nM T83011 C9Q1CD 155527777 IC50 = 22200 nM T83011 C86KIL 155527931 IC50 > 10000 nM T83011 C5Q1LN 155528022 IC50 = 3 nM T83011 CBJ75A 155528343 IC50 = 51019 nM T83011 CCU17Y 155528388 IC50 = 26900 nM T83011 CR5E7W 155528403 IC50 > 10000 nM T83011 CCA76W 155528448 IC50 > 50000 nM T83011 C4OL2X 155528461 IC50 = 10000 nM T83011 CK37ZL 155528508 IC50 = 590 nM T83011 CB17HP 155528915 IC50 = 2100 nM T83011 CQM2L6 155529262 IC50 > 50000 nM T83011 C0Q8PH 155529386 IC50 = 9352.5 nM T83011 CGX6S4 155529530 IC50 = 828 nM T83011 CM9E2L 155529630 IC50 > 200000 nM T83011 C62IFU 155529674 IC50 = 19400 nM T83011 CDT04B 155529889 IC50 = 767 nM T83011 CPOR92 155530007 IC50 = 18110 nM T83011 C7WDL3 155530036 IC50 = 932 nM T83011 CR3C2A 155530056 IC50 = 56400 nM T83011 C34VYA 155530298 IC50 > 10000 nM T83011 C4PU5G 155530390 Ki = 20.6 nM T83011 CF4JS0 155530576 IC50 = 23900 nM T83011 C1I5XU 155530592 IC50 = 480 nM T83011 CY7PE5 155530744 IC50 > 20000 nM T83011 CY3QH2 155530781 IC50 = 10000 nM T83011 C2YDZ8 155531112 IC50 > 10000 nM T83011 C5X1QC 155531135 IC50 = 802 nM T83011 C13NXZ 155531338 IC50 > 10000 nM T83011 CS35DE 155531420 IC50 > 100000 nM T83011 CEW68T 155531424 IC50 = 16700 nM T83011 CI0XL3 155531445 IC50 = 1409 nM T83011 CO1B6G 155531477 IC50 > 50000 nM T83011 C75DNP 155531484 IC50 = 8300 nM T83011 C2GH4F 155531521 IC50 = 1300 nM T83011 C92HMB 155532012 Ki = 0.57 nM T83011 CD14WR 155532205 IC50 = 285 nM T83011 CYL4B2 155532320 IC50 = 600 nM T83011 CXMC14 155532373 IC50 > 10000 nM T83011 C03YPC 155532460 IC50 = 19800 nM T83011 CD73OS 155532519 IC50 = 119300 nM T83011 CMKP85 155532627 IC50 > 50000 nM T83011 CYL4N3 155532636 Ki = 390 nM T83011 CMZ3F5 155533066 IC50 = 73 nM T83011 CE1C3L 155533414 IC50 = 335.7 nM T83011 CBL16Y 155533456 IC50 = 480 nM T83011 C31SGR 155533470 IC50 = 5200 nM T83011 CBJ65Q 155533568 IC50 = 29030 nM T83011 C8FCH7 155533611 IC50 = 723 nM T83011 C9WO1Z 155533882 IC50 = 10000 nM T83011 CN3Y7C 155534177 IC50 = 91.9 nM T83011 CKM60Q 155534231 IC50 > 10000 nM T83011 CYN5O8 155534304 IC50 = 780 nM T83011 C0R3PA 155534717 IC50 = 10000 nM T83011 CIH0T5 155535400 IC50 > 10000 nM T83011 CI40DC 155535506 IC50 > 10000 nM T83011 CZV42I 155535793 IC50 = 17690 nM T83011 CA1S4K 155535904 IC50 = 105 nM T83011 C0OGM5 155536279 IC50 = 2490 nM T83011 CLHQ12 155536307 IC50 = 15400 nM T83011 CQW8O6 155536436 IC50 = 16100 nM T83011 CLG47F 155536506 IC50 = 2070 nM T83011 C07QMN 155536709 IC50 = 26700 nM T83011 CH7C5J 155536981 IC50 = 1910 nM T83011 CMG75B 155537001 IC50 > 10000 nM T83011 C8ZG7F 155537023 IC50 = 2450 nM T83011 CP5O4N 155537289 IC50 = 3400 nM T83011 CS9M4P 155537529 IC50 = 656 nM T83011 CI5ZS1 155537565 IC50 = 145.1 nM T83011 CV39TC 155537638 IC50 = 9020 nM T83011 C5B2IG 155537846 IC50 = 424.6 nM T83011 CA6EU8 155538194 IC50 = 12700 nM T83011 CUI68E 155538243 IC50 = 59630 nM T83011 C87THM 155538450 IC50 = 1060 nM T83011 C1BHZ0 155538647 IC50 = 46 nM T83011 C6OE2W 155538683 IC50 = 21600 nM T83011 CQD2G6 155538820 IC50 = 8444.7 nM T83011 C2BQ3R 155539015 IC50 = 15200 nM T83011 C54MIG 155539279 IC50 = 3300 nM T83011 COBD26 155539285 IC50 = 630 nM T83011 C96AFW 155539339 IC50 = 215 nM T83011 CME98X 155539363 Ki = 75 nM T83011 CHVM69 155539705 IC50 = 102 nM T83011 CD9KW3 155539920 IC50 > 10000 nM T83011 CAN6Y5 155540046 IC50 = 448 nM T83011 CHL9B4 155540143 IC50 > 20000 nM T83011 CT7A3I 155540193 IC50 > 10000 nM T83011 C2K5DP 155540226 IC50 = 99.2 nM T83011 CF6ZE5 155540615 IC50 > 10000 nM T83011 C3P1ZT 155540839 IC50 = 282 nM T83011 CJ2G7I 155540870 IC50 = 94700 nM T83011 CJ4PS8 155540888 IC50 > 10000 nM T83011 C2L9TS 155540948 IC50 = 364 nM T83011 C83BZU 155540992 IC50 = 18400 nM T83011 C3MXN0 155541109 IC50 = 5100 nM T83011 CBE65T 155541185 IC50 > 10000 nM T83011 C19HQM 155541262 IC50 = 377 nM T83011 CK2DF8 155542168 IC50 = 21600 nM T83011 C7XBV5 155542241 IC50 = 52300 nM T83011 C4KWU5 155542251 IC50 = 28180 nM T83011 C76RTP 155542304 IC50 = 11130 nM T83011 CX4P8S 155542351 IC50 = 4810 nM T83011 C1Y8QV 155542382 IC50 > 20000 nM T83011 C56SIN 155542407 IC50 = 1469.5 nM T83011 CYZ0M2 155542430 IC50 = 289.9 nM T83011 CCV87Q 155542600 IC50 = 515 nM T83011 C8JY0G 155542643 IC50 = 570 nM T83011 C0H7IT 155542980 IC50 = 298 nM T83011 C9VS1J 155543043 IC50 = 104700 nM T83011 CB61AN 155543072 IC50 = 301.3 nM T83011 CMU24O 155543147 IC50 = 41110 nM T83011 CQB52M 155543548 IC50 = 11700 nM T83011 CH6M5J 155543647 IC50 = 12800 nM T83011 CC4KN9 155543685 IC50 = 65 nM T83011 CB1XH5 155544104 IC50 = 36700 nM T83011 CZ8KL6 155544230 IC50 = 248600 nM T83011 C5AE8I 155544346 IC50 = 200 nM T83011 CH1G4C 155544368 IC50 > 10000 nM T83011 C5HDZ9 155544380 IC50 = 113 nM T83011 C6YJN8 155544587 IC50 = 1900 nM T83011 C30NOS 155544777 IC50 > 1000 nM T83011 C4FK7P 155544824 IC50 = 6400 nM T83011 CO7H2E 155545357 IC50 = 3440 nM T83011 C5Y4BH 155545414 IC50 = 197 nM T83011 C7JNP0 155545476 IC50 = 3800 nM T83011 C3N2AX 155545498 IC50 = 156 nM T83011 CLB1P9 155545663 IC50 = 1100 nM T83011 C7RWG6 155545712 IC50 = 373900 nM T83011 CVF2T8 155545893 IC50 = 962 nM T83011 CP15TU 155546048 IC50 = 13800 nM T83011 C4BHE8 155546183 IC50 > 1000 nM T83011 C47KJH 155546201 IC50 = 250 nM T83011 CF4V6H 155546226 IC50 = 1700 nM T83011 C6XP3U 155546562 IC50 = 1180 nM T83011 CF01DI 155546636 IC50 = 126.5 nM T83011 C1X2GS 155546843 IC50 > 10000 nM T83011 C60OKG 155547117 IC50 = 1210 nM T83011 C9E5GH 155547187 IC50 = 3.31 nM T83011 C0MYF3 155547509 IC50 = 36.1 nM T83011 CK1X5S 155547588 IC50 = 346 nM T83011 CTSF03 155547695 IC50 = 22100 nM T83011 C42XEK 155547698 IC50 > 10000 nM T83011 C8Q7JG 155547782 IC50 = 150 nM T83011 C12EGC 155547881 IC50 = 10100 nM T83011 C0OAH3 155547969 IC50 = 79 nM T83011 CLS3W9 155548122 Ki = 3420 nM T83011 C91ODF 155548523 IC50 = 570 nM T83011 C4MIT2 155548780 IC50 = 396 nM T83011 CON2H6 155548824 IC50 = 12260 nM T83011 CW89KS 155549035 IC50 = 538 nM T83011 CAZ74H 155549176 IC50 = 4800 nM T83011 CUK96G 155549201 IC50 = 16800 nM T83011 C98ABG 155549562 IC50 = 54 nM T83011 C3M2DC 155549619 IC50 = 134200 nM T83011 CG9K3X 155549681 IC50 = 172800 nM T83011 C8NGB6 155549718 IC50 = 579 nM T83011 CY5P6K 155549919 IC50 = 568 nM T83011 CR71KX 155549981 IC50 = 33100 nM T83011 C7ARS4 155550007 IC50 = 89 nM T83011 CC45SE 155550088 IC50 = 583 nM T83011 CLB3I7 155550150 IC50 = 614 nM T83011 CS8J2W 155550156 IC50 = 1500 nM T83011 C7ZK8C 155550291 IC50 = 43670 nM T83011 C2IU1J 155550532 IC50 = 1917 nM T83011 CWL16Z 155550534 IC50 > 100000 nM T83011 CVUZ30 155550746 IC50 = 156800 nM T83011 C9CKH4 155550772 IC50 > 50000 nM T83011 CM41NQ 155550778 IC50 = 756 nM T83011 C6J5EX 155550807 IC50 = 10000 nM T83011 C1J7SD 155550841 IC50 = 445 nM T83011 CNMF93 155550975 IC50 = 4574 nM T83011 CXJM04 155551396 IC50 = 16600 nM T83011 COR5T3 155551621 IC50 > 200000 nM T83011 C8JD0O 155551671 IC50 = 9630 nM T83011 CCD10R 155551712 IC50 = 439 nM T83011 CI0WL8 155551843 IC50 = 6221.5 nM T83011 C5H0FB 155552050 IC50 = 17170 nM T83011 CA3SR7 155552282 IC50 = 14440 nM T83011 CFZ7K1 155552358 IC50 > 200000 nM T83011 C2R0DM 155552400 IC50 = 26.45 nM T83011 CM40UT 155552539 IC50 = 264 nM T83011 CIQH30 155552719 IC50 = 171 nM T83011 CT9D2Y 155553307 IC50 = 11745.1 nM T83011 C1RLI0 155553370 IC50 = 991 nM T83011 C1A5OR 155553697 IC50 = 1500 nM T83011 CB75AP 155553750 IC50 > 1000 nM T83011 CC98IO 155554016 IC50 = 12 nM T83011 CR2YV5 155554100 IC50 = 237600 nM T83011 CP10LB 155554293 IC50 = 102 nM T83011 C0F2DU 155554431 IC50 = 417 nM T83011 CNA12V 155554517 IC50 = 239 nM T83011 CSI9P4 155554561 IC50 > 100000 nM T83011 CZLJ35 155554879 IC50 = 4000 nM T83011 CT06QZ 155555033 IC50 = 120 nM T83011 CQ4X0Z 155555067 IC50 = 110 nM T83011 CQKH19 155555069 IC50 = 21980 nM T83011 CCV7X8 155555111 IC50 = 480 nM T83011 C57MKC 155555241 IC50 = 343 nM T83011 CQK21Y 155555466 IC50 = 110 nM T83011 CR97GM 155555497 IC50 = 277600 nM T83011 C4F5XM 155555673 IC50 = 1100 nM T83011 CXMC57 155555780 IC50 = 213400 nM T83011 CJ73SL 155556032 IC50 = 111000 nM T83011 C2VP0T 155556202 IC50 = 10000 nM T83011 C8UQR0 155556261 IC50 = 920 nM T83011 CJ75TC 155556370 IC50 = 10495 nM T83011 CEF72R 155556374 IC50 = 13780 nM T83011 CV9P2M 155556457 IC50 = 10000 nM T83011 CC14ON 155556524 IC50 = 310 nM T83011 CSN6O4 155556536 IC50 = 47600 nM T83011 C15AIW 155556670 IC50 = 8100 nM T83011 CNM4F3 155556727 IC50 = 2230 nM T83011 C8QW7M 155556988 IC50 = 1160 nM T83011 CGZ08K 155557025 IC50 = 155500 nM T83011 C9FG2V 155557097 IC50 = 90 nM T83011 C9MWG2 155557128 IC50 = 132 nM T83011 CV21NW 155557226 IC50 = 425 nM T83011 CTVQ18 155557424 IC50 = 20350 nM T83011 CTSX95 155557611 IC50 > 1000 nM T83011 CPV60C 155557921 Ki = 44.1 nM T83011 CJ16GB 155557960 IC50 = 275 nM T83011 COS3I5 155558121 IC50 = 1860 nM T83011 C4I5JH 155558217 IC50 = 184100 nM T83011 C0GO3J 155558260 IC50 = 27900 nM T83011 C0W7AL 155558312 IC50 > 10000 nM T83011 C3A7MK 155558447 IC50 = 1070 nM T83011 C8Z2TC 155558489 IC50 > 10000 nM T83011 C2VI9G 155558502 IC50 = 428 nM T83011 CE4B5Q 155558687 IC50 = 100000 nM T83011 CLP06Y 155558745 IC50 = 14.7 nM T83011 C0YIQ1 155558898 IC50 = 4.5 nM T83011 CFV87L 155559083 IC50 = 31.61 nM T83011 C9XQ0B 155559130 IC50 = 612 nM T83011 CTI57G 155559203 IC50 = 313 nM T83011 C2B8NX 155559219 IC50 > 10000 nM T83011 C2IE8Y 155559365 IC50 = 3700 nM T83011 CT0A9X 155559380 IC50 > 20000 nM T83011 CP87XK 155559423 IC50 > 1000 nM T83011 CW5A8X 155559793 IC50 = 23400 nM T83011 C0AI5O 155560069 IC50 = 114 nM T83011 C2KI9B 155560090 IC50 = 2640.1 nM T83011 CP3T1Z 155560136 IC50 = 24940 nM T83011 C0HB4R 155560171 IC50 = 4900 nM T83011 C1H2BO 155560312 IC50 > 50000 nM T83011 C6W7SI 155560321 IC50 = 24 nM T83011 C8B7CG 155560391 IC50 = 83 nM T83011 CA35OS 155560404 IC50 = 125.89 nM T83011 C3OP1F 155560545 IC50 = 426 nM T83011 C51KNM 155560680 IC50 = 15710 nM T83011 CXJ23G 155560844 IC50 = 17200 nM T83011 C9OR6P 155560910 IC50 = 2.65 nM T83011 CU0E7C 155561006 IC50 = 9980 nM T83011 CEXP80 155561009 IC50 = 1350 nM T83011 C6P9GA 155561569 IC50 = 39 nM T83011 CP6T9Q 155561572 IC50 = 264.9 nM T83011 C63PUA 155561583 IC50 = 3600 nM T83011 C1IA4X 155561597 IC50 > 10000 nM T83011 C5R3LT 155561606 IC50 = 1160 nM T83011 CWAG35 155561892 IC50 = 17300 nM T83011 C2JQ3C 155561938 IC50 > 50000 nM T83011 CK5G2U 155562162 IC50 = 549 nM T83011 CR06HY 155562212 IC50 = 7396 nM T83011 CUK35V 155562664 IC50 = 20120 nM T83011 C1NF2M 155562789 IC50 = 840 nM T83011 C4W2LI 155563026 IC50 = 1.73 nM T83011 C9JPF8 155563044 IC50 = 396600 nM T83011 CRN35V 155563086 IC50 = 18700 nM T83011 CM46KC 155563177 IC50 > 1000 nM T83011 CQ19VC 155563189 IC50 = 991 nM T83011 CA27NL 155563199 IC50 > 10000 nM T83011 CK0EO8 155563307 IC50 = 7411.6 nM T83011 CS85JQ 155563497 IC50 = 39700 nM T83011 C26SAU 155563561 IC50 = 9500 nM T83011 CPTM25 155563673 IC50 = 407 nM T83011 C5ZKN0 155563788 IC50 > 1000 nM T83011 CD6QW7 155563833 IC50 = 2130 nM T83011 C2IGH8 155563922 IC50 = 10700 nM T83011 CZ6PB4 155564063 IC50 = 2038 nM T83011 COF96P 155564105 IC50 > 100000 nM T83011 C6U4XC 155564123 IC50 = 17200 nM T83011 CE2V5Y 155564179 IC50 = 177 nM T83011 CV6XI3 155564440 IC50 = 736 nM T83011 CY6OR7 155564797 IC50 = 550 nM T83011 C83BSZ 155564858 IC50 = 190500 nM T83011 CL09BS 155565080 IC50 = 15700 nM T83011 CUA4I7 155565084 IC50 = 65000 nM T83011 CVY9L7 155565232 IC50 = 975 nM T83011 CKGC67 155565439 IC50 > 10000 nM T83011 CJ0W5N 155565612 IC50 = 2600 nM T83011 CQJ2G8 155565621 IC50 = 192.6 nM T83011 C8N3PQ 155565636 IC50 = 371 nM T83011 CYI54E 155565672 IC50 > 1000 nM T83011 CI2CQ0 155565683 IC50 = 411 nM T83011 C8NMH4 155565767 IC50 = 25800 nM T83011 CE04NW 155566969 IC50 = 3100 nM T83011 C8OL6E 155567040 IC50 = 1900 nM T83011 CS7D2L 155567545 IC50 = 427 nM T83011 C7GU2Y 155568113 IC50 = 270 nM T83011 CKPH62 155568351 IC50 = 1.023 nM T83011 CS6K7G 155568564 IC50 = 23440 nM T83011 CK94OC 155568569 IC50 = 3100 nM T83011 C3X5ML 155568799 IC50 = 9230 nM T83011 C8S0FZ 155568919 IC50 = 49510 nM T83011 CPUO78 155569044 IC50 = 20800 nM T83011 CH86AJ 155569073 IC50 = 758 nM T83011 CZC4R7 155569133 IC50 = 1506.6 nM T83011 C0MSD7 155569179 IC50 = 2195.6 nM T83011 CQ1LV7 135508617 IC50 = 2700 nM T83011 CGK7B1 135511529 IC50 = 43167 nM T83011 CRKP76 136016509 IC50 = 24500 nM T83011 D00AVR 135476741 IC50 = 10017 nM T83011 D00HVZ 5271544 IC50 = 7180 nM T83011 D00OLX 46232855 Ki = 140 nM T83011 D00OQL 3852139 IC50 = 165 nM T83011 D00PJT 46232080 IC50 = 150 nM T83011 D00RIX 5280443 IC50 = 12800 nM T83011 D00RNZ 910172 IC50 = 1.698 nM T83011 D00WSM 599289 IC50 = 600 nM T83011 D00WVG 584447 IC50 = 296 nM T83011 D01GAX 1388 Ki = 280000 nM T83011 D01HQV 45485414 IC50 = 155.59 nM T83011 D01KZF 46232145 IC50 = 160 nM T83011 D01LUB 4297278 IC50 = 3870 nM T83011 D01UFM 724217 IC50 = 500 nM T83011 D01VPZ 15352647 IC50 = 6690 nM T83011 D02AQM 6918822 IC50 = 1500 nM T83011 D02FJX 46232854 Ki = 1300 nM T83011 D02KGZ 10657190 IC50 = 7680 nM T83011 D02KXU 15098246 IC50 = 550 nM T83011 D02WOQ 46232079 IC50 = 150 nM T83011 D02ZZA 44424447 Ki > 100000 nM T83011 D03BQJ 688829 IC50 = 2380 nM T83011 D03EPY 7046 Ki = 15000 nM T83011 D03LGV 11241513 IC50 = 3700 nM T83011 D03PXS 341782 IC50 = 760 nM T83011 D03XQB 5271543 IC50 = 170 nM T83011 D04DCW 46231665 IC50 = 130 nM T83011 D04FLL 20242416 Ki > 100000 nM T83011 D04LPY 46232853 Ki = 370 nM T83011 D04TGN 181620 IC50 = 48 nM T83011 D04TZI 12098585 IC50 = 19000 nM T83011 D05CCT 4139 IC50 = 4370 nM T83011 D05ODW 91510 Ki = 54 nM T83011 D05QOR 5280460 IC50 > 60000 nM T83011 D05WQN 46400456 Ki = 3000 nM T83011 D06AAA 11390419 IC50 = 4800 nM T83011 D06AJP 44575103 Ki = 1400 nM T83011 D06ERH 637760 IC50 = 1412537.54 nM T83011 D06QNN 120587 IC50 = 1960 nM T83011 D07BAO 5289289 Ki = 17000 nM T83011 D07GUX 42629116 Ki = 266 nM T83011 D07HFF 46232008 IC50 = 7610 nM T83011 D07NBB 46232852 Ki = 68 nM T83011 D07TAJ 914298 IC50 = 23460 nM T83011 D07WFU 44577750 IC50 = 20000 nM T83011 D07WIJ 46232077 IC50 = 150 nM T83011 D08CNS 3748 IC50 = 7.54 nM T83011 D08FFH 701943 IC50 = 17300 nM T83011 D08FXH 46233267 Ki = 130 nM T83011 D08HKC 46232005 IC50 = 6720 nM T83011 D08ILX 24219274 Ki = 1650 nM T83011 D08NQM 5289247 IC50 = 13000 nM T83011 D08PHY 11171752 IC50 = 4900 nM T83011 D08SSS 44424448 Ki = 14030 nM T83011 D08TFN 4996817 Ki > 100000 nM T83011 D08YCE 46232851 Ki = 230 nM T83011 D09FAD 823440 IC50 = 3270 nM T83011 D09HBX 10374615 IC50 = 6400 nM T83011 D09NNZ 46947643 Ki = 30 nM T83011 D09PBW 46232075 IC50 = 650 nM T83011 D09XSB 42628986 Ki = 4 nM T83011 D0A1RE 44407281 IC50 = 5570 nM T83011 D0A2AF 5289295 Ki = 600 nM T83011 D0A2FO 2825024 IC50 = 1470 nM T83011 D0A4IY 5196 IC50 = 6.7 nM T83011 D0B1WD 724200 IC50 = 890 nM T83011 D0B1XZ 15731432 IC50 = 170 nM T83011 D0B2TV 44577747 IC50 = 18000 nM T83011 D0B3QN 46232081 IC50 = 140 nM T83011 D0B6MV 658198 Ki = 1100 nM T83011 D0BV8Y 179342 IC50 = 0.9 nM T83011 D0C1LI 53378764 IC50 = 39 nM T83011 D0C9GI 46231795 IC50 = 4330 nM T83011 D0C9WW 16750123 Ki = 400 nM T83011 D0D2JH 46231663 IC50 = 670 nM T83011 D0D5KD 46233198 Ki = 16900 nM T83011 D0D6OR 46233269 Ki = 38 nM T83011 D0D6QI 24219273 Ki = 330 nM T83011 D0DQ6Z 8530 Ki = 1500 nM T83011 D0E4HB 8443728 IC50 = 116 nM T83011 D0E8IE 3110315 IC50 = 1140 nM T83011 D0F2DC 11816512 IC50 = 13000 nM T83011 D0F2SM 46232144 IC50 = 200 nM T83011 D0F3VE 379338 IC50 = 74.13 nM T83011 D0F7KG 2329349 IC50 = 195 nM T83011 D0G3BI 25090 IC50 = 19.05 nM T83011 D0G6MA 10378415 IC50 = 5140 nM T83011 D0GN5Z 5281295 IC50 > 80000 nM T83011 D0H0GZ 599290 IC50 = 710 nM T83011 D0H1VT 11423691 IC50 = 37000 nM T83011 D0H3NS 10752 IC50 = 17.38 nM T83011 D0H3RQ 46933990 IC50 = 3230 nM T83011 D0HU4J 5004199 Ki > 100000 nM T83011 D0I2GP 50876172 IC50 = 1096.48 nM T83011 D0I3XA 6422124 IC50 = 1900 nM T83011 D0I5CZ 46232076 IC50 = 620 nM T83011 D0I9AA 46231936 IC50 = 1610 nM T83011 D0IA3U 44442376 IC50 = 223.87 nM T83011 D0ID3Y 46233197 Ki > 100000 nM T83011 D0IK2S 5270543 IC50 = 3770 nM T83011 D0J0MX 641683 Ki = 0.6 nM T83011 D0J0QW 46233266 Ki = 2100 nM T83011 D0J2UA 135433933 IC50 = 447 nM T83011 D0JN9R 223566 Ki = 430 nM T83011 D0K1FE 46933989 IC50 = 11050 nM T83011 D0K5LJ 5289310 IC50 = 14 nM T83011 D0K8EE 261394 IC50 = 12940 nM T83011 D0L6HE 46232078 IC50 = 170 nM T83011 D0LI3J 3080926 Ki = 8300 nM T83011 D0M2EM 4650 IC50 = 10200 nM T83011 D0M4GR 46233264 Ki = 460 nM T83011 D0M7BR 5280378 IC50 = 25800 nM T83011 D0M8UY 72139 IC50 = 9570 nM T83011 D0N4DR 46232141 IC50 = 110 nM T83011 D0NS1S 5280442 Ki = 49 nM T83011 D0O0MY 15462540 IC50 = 3350 nM T83011 D0O1GE 44622873 IC50 = 0.8 nM T83011 D0P1YC 46232142 IC50 = 530 nM T83011 D0P4GF 25139469 IC50 = 1.49 nM T83011 D0P7SY 1231330 IC50 = 480 nM T83011 D0Q1IP 5273551 IC50 = 27.54 nM T83011 D0R3LP 2802466 IC50 = 2070 nM T83011 D0R6FJ 64961 Ki = 1120 nM T83011 D0R9TX 14054762 IC50 = 13.05 nM T83011 D0S0JH 44563082 IC50 = 16530 nM T83011 D0SP2O 7054 Ki = 33 nM T83011 D0T1GP 12549536 IC50 = 3620 nM T83011 D0T1YO 379337 IC50 = 177.83 nM T83011 D0T3XC 46233268 Ki = 68 nM T83011 D0T3ZS 46233265 Ki = 48 nM T83011 D0T7VA 102928 IC50 = 2200 nM T83011 D0T9ZL 2703 IC50 > 20000 nM T83011 D0TB1E 46232143 IC50 = 590 nM T83011 D0TL3S 25139473 IC50 = 9360 nM T83011 D0TU7I 5353365 IC50 = 17.8 nM T83011 D0U8ET 49864488 IC50 = 4300 nM T83011 D0UL6Y 11401479 IC50 = 10000 nM T83011 D0US0J 5961410 IC50 = 18620871.37 nM T83011 D0V3NT 34521 Ki = 15000 nM T83011 D0V6DF 11615193 IC50 = 71000 nM T83011 D0VB2W 21501 IC50 = 2500 nM T83011 D0W1WE 16376796 IC50 = 8890 nM T83011 D0W7XK 466270 IC50 = 1340 nM T83011 D0X8HH 44575104 Ki = 600 nM T83011 D0X8RN 6971118 IC50 = 19000 nM T83011 D0XJ7I 6683 IC50 > 40000 nM T83011 D0Y0KU 46231664 IC50 = 160 nM T83011 D0Y1XS 701990 IC50 = 28130 nM T83011 D0Y4SO 46223113 IC50 > 150000 nM T83011 D0Y5OB 46231935 IC50 = 6890 nM T83011 D0Y7HG 5281616 IC50 = 3650 nM T83011 D0Y8AN 5195 IC50 = 19.6 nM T83011 D0Z0ZU 23661626 Ki = 4580 nM T83011 D0Z2XR 46231666 IC50 = 500 nM T83011 D0Z5BU 46233199 Ki = 2400 nM T83011 D0ZH0T 11032058 IC50 = 4410 nM T83011 D0ZI0S 930709 IC50 = 11340 nM T15882 D0FT4R 107706 IC50 = 340 nM T15882 CC9E0Y 232547 IC50 = 12800 nM T15882 CF9VK2 5236960 IC50 > 139000 nM T15882 C63HAE 18572952 IC50 > 134000 nM T15882 CN0VA7 24822701 IC50 > 50000 nM T15882 C3GS6F 33009902 IC50 > 10000 nM T15882 C96CKU 49797573 IC50 > 50000 nM T15882 C48UHX 66561877 IC50 = 14500 nM T15882 C1MBU7 72793747 IC50 = 5900 nM T15882 C6BY5D 72793776 IC50 = 47500 nM T15882 C1DI8A 72793778 IC50 > 100000 nM T15882 CHO59P 101883943 IC50 = 530 nM T15882 C8E4WS 102323332 IC50 > 50000 nM T15882 CR2AU7 118010068 IC50 = 610 nM T15882 COA36C 118010069 IC50 = 2370 nM T15882 C5NJH1 118202505 IC50 = 2500 nM T15882 C43ADS 118202506 IC50 = 470 nM T15882 C2UXT7 118202507 IC50 = 220 nM T15882 CPV27G 118202509 IC50 = 2050 nM T15882 CJB3K7 118202510 IC50 = 1090 nM T15882 C12BHL 118202511 IC50 = 1730 nM T15882 COT6H0 118202512 IC50 = 360 nM T15882 C5FU4E 118723831 IC50 = 10380 nM T15882 C8ZSC2 118727248 IC50 = 2310 nM T15882 CYIX41 118727249 IC50 = 530 nM T15882 CH1T3M 118727250 IC50 = 2050 nM T15882 CVG1X5 118727251 IC50 = 3020 nM T15882 C9B6KX 118727252 IC50 = 3910 nM T15882 C3OUW6 118727253 IC50 > 10000 nM T15882 C10QJC 118727254 IC50 > 10000 nM T15882 CVIF56 118727255 IC50 > 10000 nM T15882 CNQ9U4 118727256 IC50 = 4940 nM T15882 CN93WU 118727257 IC50 > 10000 nM T15882 C5DR7Z 118727258 IC50 > 10000 nM T15882 CDEU05 118727259 IC50 = 310 nM T15882 CZHT12 118727260 IC50 = 610 nM T15882 CNL2Z9 137635679 Ki > 10000 nM T15882 C6V7PE 137638228 Ki = 5.4 nM T15882 C03IMN 137647139 Ki > 10000 nM T15882 C7BY8N 137647576 Ki = 21 nM T15882 CZ1H4R 137655362 Ki > 10000 nM T15882 CP2V3H 137656873 Ki = 3600 nM T15882 CTUM82 137658421 IC50 = 54000 nM T15882 CBU5W0 155524880 Ki = 17 nM T15882 C8U9ED 155533652 Ki = 245 nM T15882 C93MCB 155534384 Ki = 51 nM T15882 CLRB54 155544531 Ki = 9.8 nM T15882 C2E5GR 155554478 Ki = 7 nM T15882 CFX07G 155558369 Ki = 6.1 nM T15882 CVB89F 155568340 Ki = 23 nM T15882 D0C1NP 66561876 IC50 = 1400 nM T15882 D0S5RY 4784 IC50 = 19230 nM T72024 C1EH0P 501640 IC50 > 30000 nM T72024 C1MD8E 145981653 IC50 > 30000 nM T72024 CP2VA7 145991605 IC50 > 30000 nM T87686 D06IAR 60961 IC50 = 100000 nM T87686 D0C6GK 57345410 Ki = 0.012 nM T87686 CZ5DA1 11824 IC50 = 44000 nM T87686 CJ0I1N 13792 IC50 = 170 nM T87686 CW02OU 14978 IC50 = 26000 nM T87686 C5Q7PG 97297 IC50 = 18000 nM T87686 C5IO2D 171251 Ki = 100000 nM T87686 CA6J0D 445762 Ki = 25000 nM T87686 CP7L0Q 446940 IC50 = 22000 nM T87686 CBF5V6 470024 IC50 = 200000 nM T87686 C8VO2Q 666637 IC50 = 19390 nM T87686 CQEF34 1002773 IC50 > 100000 nM T87686 CS24EJ 1234053 IC50 = 26780 nM T87686 CUYO65 1478384 IC50 = 320000 nM T87686 CD9QW2 1972282 IC50 = 64150 nM T87686 CLKC18 1977548 IC50 = 4640 nM T87686 C4EWN3 2030255 IC50 = 8290 nM T87686 CMB25K 2231443 IC50 = 8400 nM T87686 C3V5FW 2743649 IC50 = 14000 nM T87686 C4XLM0 2992271 IC50 = 3960 nM T87686 C4L0WX 3159434 IC50 = 17370 nM T87686 CS86UD 4909931 IC50 = 4480 nM T87686 CV3X9P 5238298 IC50 = 8500 nM T87686 CSQ72Y 5311816 IC50 = 13660 nM T87686 C6V5EO 6226054 IC50 = 9410 nM T87686 C7F4PU 6226661 IC50 = 20940 nM T87686 CEN4X3 7313645 IC50 = 9700 nM T87686 C2BV1T 9836890 Ki > 100000 nM T87686 CS7QJ4 9862185 Ki > 100000 nM T87686 CSB2F9 10344836 Ki = 1100 nM T87686 CI3OG1 10916869 Ki = 2000 nM T87686 C2Y7VH 11123068 Ki = 2800 nM T87686 CDG2H3 11277569 IC50 = 200000 nM T87686 C7VG6J 11761979 Ki = 7800 nM T87686 CV29SR 11859064 IC50 = 16000 nM T87686 CMJ91K 22180707 IC50 > 100000 nM T87686 C21XVI 22180710 IC50 > 100000 nM T87686 CZEW86 22180716 IC50 > 100000 nM T87686 CKJR10 24764113 Ki > 100000 nM T87686 CB28LP 25164116 IC50 = 1500 nM T87686 C7A2EF 44121153 IC50 = 7010 nM T87686 C8F2NX 44401736 Ki > 100000 nM T87686 C9K1QF 49784135 IC50 = 41000 nM T87686 C02ORV 53377508 Ki = 290 nM T87686 CPL71I 54596764 IC50 > 100000 nM T87686 C3SX2U 56642704 IC50 = 38 nM T87686 C72GHW 56642706 IC50 = 120 nM T87686 CS6Q7R 56642708 IC50 = 110 nM T87686 C0R4GZ 56835775 Ki > 100000 nM T87686 CJBY70 56951879 Ki = 0.46 nM T87686 CKB82D 57384118 Ki = 13 nM T87686 C60IAQ 58619539 IC50 > 100000 nM T87686 CB30IV 60074592 Ki > 100000 nM T87686 C37QSD 67066693 IC50 = 251188.64 nM T87686 CER5F1 67466175 IC50 > 100000 nM T87686 CN0KD1 67973918 Ki = 70 nM T87686 C5QE6A 67988955 IC50 < 100 nM T87686 CACQ63 70675983 Ki = 690 nM T87686 CG1MQ0 70675984 Ki = 130 nM T87686 C04ANP 70675985 Ki = 1000 nM T87686 CN74VL 70675986 Ki = 80 nM T87686 CSIJ50 70675987 Ki = 2700 nM T87686 C8JTS3 70676140 Ki = 0.76 nM T87686 CZL47S 70676141 Ki = 12 nM T87686 C8KC6O 70676142 Ki = 22 nM T87686 C9QH8N 70677532 Ki > 100000 nM T87686 C8RLI4 70677678 Ki > 100000 nM T87686 C7BZ6R 70677679 Ki > 100000 nM T87686 CRW2L0 70677680 Ki > 100000 nM T87686 CP3QD9 70677681 Ki > 100000 nM T87686 CED83W 70677682 Ki = 50000 nM T87686 C39DOF 70677683 Ki = 46000 nM T87686 CBH29R 70677811 Ki = 47000 nM T87686 C8IWP5 70677812 Ki > 100000 nM T87686 C2U0SD 70677813 Ki = 22000 nM T87686 CQE8F1 70677814 Ki > 100000 nM T87686 C5JUD8 70677815 Ki > 100000 nM T87686 C1O2FI 70677816 Ki > 100000 nM T87686 C6G9XO 70677960 Ki = 22000 nM T87686 C5EJU1 70677961 Ki = 16000 nM T87686 CZ0GF8 70677962 Ki = 1900 nM T87686 COJF34 70677963 Ki = 5500 nM T87686 C5NJ2L 70677964 Ki = 17000 nM T87686 CPY19A 70677965 Ki = 4500 nM T87686 CQW50G 70678103 Ki = 550 nM T87686 CVR7U8 70678104 Ki = 18000 nM T87686 C5N2XS 70678105 Ki = 1100 nM T87686 CI9TH5 70678106 Ki = 350 nM T87686 C30BZK 70678107 Ki = 70 nM T87686 C95RGA 70678245 Ki = 82 nM T87686 C5BD3O 70678246 Ki = 190 nM T87686 C04YNM 70678247 Ki = 270 nM T87686 C7UQ6V 70678248 Ki = 58 nM T87686 CYJ92K 70678249 Ki = 140 nM T87686 CP5C1T 71405007 Ki = 12000 nM T87686 CUCB21 71449865 Ki = 6500 nM T87686 CPR79J 71449866 Ki = 8900 nM T87686 C6MR3G 71457019 Ki = 2000 nM T87686 C06TQH 71460688 Ki = 3800 nM T87686 CUP4Q6 76328021 Ki = 1.3 nM T87686 CX7V5M 76328022 Ki = 1.1 nM T87686 CHBY56 76328033 Ki = 20000 nM T87686 CZH43W 76331386 IC50 = 1080 nM T87686 C5P2BM 76331683 Ki > 50000 nM T87686 C4XJ5N 78357767 IC50 > 100000 nM T87686 CT82JP 115790497 IC50 = 139000 nM T87686 CFC42D 118735770 IC50 = 99000 nM T87686 CMHZ30 118735771 IC50 > 100000 nM T87686 CSB1V0 118735772 IC50 > 100000 nM T87686 C0O9KV 121005803 IC50 = 4400 nM T87686 C6K1NE 121005804 IC50 = 20 nM T87686 C7PRI3 121005805 IC50 = 10 nM T87686 C5FB7C 121005806 IC50 = 150 nM T87686 CC1AN3 121005807 IC50 = 39000 nM T87686 CV0FW8 121225442 IC50 = 13 nM T87686 C2PF1E 121231410 Ki = 0.08 nM T87686 C3OFP2 124222436 Ki = 0.002 nM T87686 CNO7R6 133364127 IC50 = 4600 nM T87686 CF29KH 134159782 IC50 = 1300 nM T87686 CF5M8D 137633763 IC50 = 4 nM T87686 CDB81C 137642264 IC50 = 3.981 nM T87686 CVG0X6 137646229 IC50 = 0.15 nM T87686 CN2U8J 137647431 IC50 = 1430 nM T87686 C9WA0R 137650875 IC50 = 6.34 nM T87686 CGLK72 137652671 IC50 = 690 nM T87686 CVZ98H 137654322 IC50 = 7943.28 nM T87686 C4D9ZU 137655088 IC50 = 141000 nM T87686 C31VTO 137662130 IC50 = 2160 nM T87686 C8LEV4 139267760 IC50 > 10000 nM T87686 C4KJG0 145704694 IC50 = 270 nM T87686 C0UB2Z 145704695 IC50 = 0.11 nM T87686 C60XTA 145704696 IC50 = 0.17 nM T87686 CX08EA 145712402 IC50 = 0.19 nM T87686 C56JFR 145993747 IC50 = 96000 nM T87686 CD28UO 146680921 IC50 = 14 nM T87686 CS4Q9C 155510713 IC50 = 98000 nM T87686 CD7HB9 155512163 IC50 = 47 nM T87686 CNLT34 155518616 IC50 = 840 nM T87686 CF0D7W 155519587 IC50 = 2.1 nM T87686 C6Y5ML 155523008 IC50 = 21670 nM T87686 C1MB6D 155526865 IC50 = 4350 nM T87686 CA6BL8 155537337 IC50 = 920 nM T87686 CJDY13 155539676 IC50 = 1060 nM T87686 C5ZQW4 155543019 IC50 = 43000 nM T87686 CI0O3G 155546745 Ki = 0.36 nM T87686 CD7JN0 155546855 IC50 = 4100 nM T87686 CY1C7G 155547867 IC50 = 1100 nM T87686 CUY45S 155549063 IC50 = 89 nM T87686 C2J4QN 155554452 IC50 = 28000 nM T87686 CV78BF 155554518 IC50 = 0.59 nM T87686 C0MFL7 155558010 IC50 = 28.2 nM T87686 C4BAZ8 155559544 IC50 = 22800 nM T87686 CIU2H8 155563241 IC50 = 280 nM T87686 C50XOL 155563966 IC50 = 4300 nM T87686 CR78JU 155566532 IC50 = 4300 nM T87686 C90WDC 155566570 IC50 = 97 nM T87686 CJIC70 155567955 IC50 = 16 nM T87686 C25MSB 155568468 IC50 = 40000 nM T87686 D00FLT 65482 IC50 = 33710 nM T87686 D02TVQ 71268957 IC50 > 100000 nM T87686 D03OLX 25231309 Ki = 9000 nM T87686 D09CLP 439155 Ki = 160 nM T87686 D09ENZ 56962336 Ki = 0.3 nM T87686 D0L0DC 53339032 Ki = 38 nM T87686 D0S9SJ 56962337 EC50 = 9 nM T63179 D04DJN 10635 IC50 = 360 nM T63179 D07BSQ 5994 IC50 = 14 nM T63179 D0D1SG 5755 EC50 = 0.002 nM T63179 D0EP0C 5833 IC50 = 1.6 nM T63179 D0G8BV 6450278 Ki = 37 nM T63179 D0I1LH 5839 EC50 = 0.18 nM T63179 D0IT2G 5743 Ki = 0.36 nM T63179 D0Q4SD 443872 IC50 = 63.1 nM T63179 D0Y7IU 5281004 EC50 = 4.8 nM T63179 D0Y7JU 9854489 IC50 = 166 nM T63179 D0Z4EI 55245 IC50 = 590 nM T63179 D00JFE 56941241 IC50 > 1000 nM T63179 D01SYU 10026128 IC50 = 10000 nM T63179 D05RZE 42636651 Ki = 0.33 nM T63179 D07MON 5311505 IC50 = 470 nM T63179 D0SZ1G 121248172 IC50 > 38000 nM T63179 D0X9YP 67041274 IC50 > 10000 nM T63179 D0TH6M 25204767 EC50 > 10000 nM T63179 D0W1XE 91827457 IC50 > 10000 nM T63179 D02KAU 46871935 IC50 = 9 nM T63179 D03KTE 16750192 Ki > 10000 nM T63179 D09UFV 24825740 IC50 > 5000 nM T63179 D0W5RL 9577221 IC50 = 1600 nM T63179 C59UQE 6279 IC50 = 1197 nM T63179 C2O8KM 101788 EC50 = 50 nM T63179 C40YBS 444036 IC50 = 149 nM T63179 C8AMD7 2848661 IC50 = 460 nM T63179 CLBV35 3699263 IC50 = 850 nM T63179 C43BVE 3816305 IC50 = 1070 nM T63179 CDCK27 5185174 IC50 = 1400 nM T63179 C16ZSG 6439929 Ki = 39 nM T63179 C7REX1 9805004 IC50 = 38 nM T63179 CV87EA 9820084 IC50 = 290 nM T63179 C8A3WG 9820510 Ki > 10000 nM T63179 C06RXB 9821393 Ki = 1682 nM T63179 CD9S5P 9825465 Ki = 3838 nM T63179 CE62WD 9839013 IC50 > 1000 nM T63179 CBS8M2 9839134 IC50 = 2369 nM T63179 C92CPK 9841404 Ki > 10000 nM T63179 CK7UC3 9841413 Ki > 10000 nM T63179 C7P6XH 9842832 Ki > 10000 nM T63179 C7RS9U 9846657 Ki > 5000 nM T63179 CERF28 9861044 Ki > 10000 nM T63179 C3K4EU 9862027 Ki > 10000 nM T63179 CEM27C 9885473 IC50 = 3000 nM T63179 C6B9CZ 9888873 IC50 = 160 nM T63179 CZ5R9B 9890023 Ki = 493 nM T63179 CJ7U3R 9904286 IC50 > 10000 nM T63179 C6SWK1 9904610 IC50 = 2492 nM T63179 CTI1J8 9905296 Ki > 10000 nM T63179 CE1TK2 9908041 IC50 > 10000 nM T63179 CMJG42 9921530 IC50 > 10000 nM T63179 C39EXP 9933936 IC50 = 454 nM T63179 C24FUO 9943699 IC50 = 1386 nM T63179 CCSX75 9949772 IC50 = 1500 nM T63179 CKU64T 9952569 IC50 = 333 nM T63179 CW0ED9 9953456 IC50 = 681 nM T63179 C95CAN 9978625 Ki = 0.967 nM T63179 C1QP8T 9993897 IC50 = 2000 nM T63179 C4V6RF 9998996 IC50 > 5000 nM T63179 CC4WY6 10024990 IC50 = 1000 nM T63179 CSM0W3 10026120 IC50 > 2000 nM T63179 CFY67M 10070808 IC50 = 2219 nM T63179 C9T4HR 10071810 IC50 = 1100 nM T63179 CQ3LD1 10091351 IC50 = 1600 nM T63179 C16HAK 10094808 IC50 > 2000 nM T63179 CR0DX5 10126475 IC50 > 1130 nM T63179 CHS18G 10126476 IC50 > 2000 nM T63179 CR0BP6 10126871 IC50 = 380 nM T63179 CV5PQ0 10126940 IC50 = 500 nM T63179 CVF40M 10127159 IC50 = 350 nM T63179 C3CRZ1 10127269 IC50 = 450 nM T63179 CPB60D 10127340 IC50 = 760 nM T63179 CKMW98 10128037 IC50 = 585 nM T63179 C1GI3D 10150743 IC50 = 220 nM T63179 CZKF71 10150825 IC50 = 400 nM T63179 CYR0U5 10150851 IC50 > 2000 nM T63179 CVO1F7 10151165 IC50 = 405 nM T63179 C6EC1P 10151186 IC50 = 405 nM T63179 CQ14RM 10151357 IC50 = 535 nM T63179 CW4Y2K 10151995 IC50 = 1650 nM T63179 C0MX7K 10157532 IC50 = 893 nM T63179 CL0U4N 10172897 IC50 = 400 nM T63179 CG0VH8 10173354 IC50 = 1250 nM T63179 CU6D8W 10173525 IC50 = 170 nM T63179 C8L7HJ 10179031 IC50 = 683 nM T63179 C41YRZ 10194268 IC50 > 740 nM T63179 CX4F7Z 10194607 IC50 > 2000 nM T63179 CV0LE4 10194889 IC50 > 1000 nM T63179 C3O7WH 10215978 IC50 = 1350 nM T63179 C1SG4N 10216152 IC50 > 1420 nM T63179 CD0YT7 10216465 IC50 = 940 nM T63179 C1FGX9 10216535 IC50 = 415 nM T63179 CW7QX2 10216536 IC50 = 720 nM T63179 CG9OH4 10216697 IC50 = 1050 nM T63179 CXN4W1 10216788 IC50 = 1100 nM T63179 CUGN98 10217411 IC50 = 910 nM T63179 CJ9BE0 10222329 IC50 = 651 nM T63179 C84SRT 10223610 IC50 = 2154 nM T63179 CUYO17 10237223 IC50 > 1300 nM T63179 CWYK62 10238100 IC50 = 435 nM T63179 C1R8GY 10238297 IC50 = 900 nM T63179 CNB1V3 10238624 IC50 = 190 nM T63179 CPGF94 10238831 IC50 > 2000 nM T63179 C2AZH1 10238961 IC50 = 175 nM T63179 CSA4R3 10252455 IC50 > 2000 nM T63179 C7EGH2 10252527 IC50 = 120 nM T63179 CR59SC 10271193 IC50 = 22897 nM T63179 CPIS57 10271557 IC50 = 2252 nM T63179 CUQC81 10287415 IC50 > 1000 nM T63179 C5RC7X 10287444 IC50 = 510 nM T63179 CJT2G8 10287863 IC50 = 1400 nM T63179 C1M6WY 10288006 IC50 = 320 nM T63179 CO6UP3 10288155 IC50 = 875 nM T63179 C6C2IK 10288565 IC50 = 195 nM T63179 CNEO49 10289020 IC50 = 104 nM T63179 CLJU03 10298892 Ki = 3914 nM T63179 C9UYG8 10309447 IC50 > 1050 nM T63179 C8FM2D 10309755 IC50 = 1800 nM T63179 C1OV7M 10309756 IC50 = 715 nM T63179 C9TI4A 10310063 IC50 = 1035 nM T63179 CP9AE0 10310476 IC50 > 512 nM T63179 CV52EN 10310809 IC50 = 140 nM T63179 CR1L5N 10311251 IC50 = 104 nM T63179 CX7WS4 10316069 IC50 = 354 nM T63179 CQP1Y7 10340204 IC50 = 1525 nM T63179 CEJ78I 10365592 IC50 > 2000 nM T63179 CDBZ06 10372181 IC50 = 120 nM T63179 C14AIB 10384345 IC50 = 970 nM T63179 CZ5CJ3 10423330 IC50 > 10000 nM T63179 C5I3BG 10428464 Ki = 12 nM T63179 C1KE6C 10446402 IC50 = 2050 nM T63179 C0NT9D 10454007 IC50 > 5000 nM T63179 C85RBN 10474264 IC50 > 2000 nM T63179 CUL8O4 10475384 IC50 > 5000 nM T63179 CPX65M 10477088 IC50 = 130 nM T63179 C5AP6C 10503520 IC50 > 10000 nM T63179 CBEC38 10596252 IC50 = 1000 nM T63179 CC8T7J 10598305 IC50 = 1062 nM T63179 CO3V0S 10622594 IC50 = 977 nM T63179 C02ZMG 10643956 IC50 = 748 nM T63179 CYNG45 10668755 IC50 > 10000 nM T63179 CYRQ10 10691647 Ki = 1100 nM T63179 CVD2Y9 10717098 IC50 > 10000 nM T63179 CAT1X8 10741366 IC50 = 1068 nM T63179 CB3JD0 10763832 IC50 = 1358 nM T63179 C07BOR 10787258 IC50 = 2035 nM T63179 C1CRQ5 10811045 IC50 > 10000 nM T63179 CN1H5Z 10832792 IC50 = 1592 nM T63179 CHU9A4 10873317 IC50 = 334 nM T63179 CHU10G 10960295 IC50 = 1850 nM T63179 C6LYG7 11090322 IC50 > 1000 nM T63179 CXS6J7 11155441 Ki = 10 nM T63179 CQUV78 11176984 IC50 = 23 nM T63179 CL97OU 11212803 IC50 = 540 nM T63179 C4U0DF 11213029 Ki = 980 nM T63179 CRN4V2 11232136 IC50 > 3000 nM T63179 C8XPZ4 11269445 IC50 > 2000 nM T63179 C4HNB8 11269886 IC50 = 1050 nM T63179 CC0XI4 11279959 IC50 = 440 nM T63179 C4SC0W 11281576 IC50 > 5000 nM T63179 C8YL6K 11282486 IC50 = 1700 nM T63179 CUX0S2 11282904 Ki = 21 nM T63179 CIY9H5 11291999 IC50 = 1800 nM T63179 C0IQ9K 11304445 IC50 = 160 nM T63179 C0XUF2 11305564 IC50 > 5000 nM T63179 CXC9G3 11327341 IC50 > 2000 nM T63179 CT9Y4O 11339440 IC50 = 2300 nM T63179 C8FQ9B 11375180 IC50 = 21000 nM T63179 CP2DL0 11377050 IC50 = 1000 nM T63179 C76VYN 11382721 IC50 > 2000 nM T63179 CV4RO2 11384310 IC50 = 48 nM T63179 CXW40M 11384346 IC50 > 2000 nM T63179 CU7IE0 11410199 IC50 = 690 nM T63179 CO20QH 11416730 IC50 = 155 nM T63179 C5WO0U 11429662 IC50 > 5000 nM T63179 CD2Q3F 11474917 IC50 = 83 nM T63179 CC75NQ 11477616 Ki = 430 nM T63179 CQ62KS 11485693 IC50 > 3000 nM T63179 C9Q1NY 11494167 Ki = 32 nM T63179 CFLQ08 11495227 IC50 = 320 nM T63179 C03NYX 11495549 IC50 = 90 nM T63179 CR40IH 11516847 IC50 = 1800 nM T63179 CP4F8X 11517412 IC50 = 280 nM T63179 C2PB6Z 11530605 Ki = 930 nM T63179 C1R6DC 11531942 IC50 = 140 nM T63179 CZ1HA3 11538472 IC50 = 615 nM T63179 CFC1Z4 11538799 IC50 = 1100 nM T63179 CBK60G 11559947 IC50 > 2000 nM T63179 C1D9YS 11560003 IC50 > 2000 nM T63179 CB37YF 11566981 Ki = 145 nM T63179 C8WJ2F 11567609 IC50 = 780 nM T63179 C0SCT6 11588584 IC50 = 810 nM T63179 C3MW1D 11589982 IC50 = 220 nM T63179 C03QYZ 11590471 IC50 = 110 nM T63179 CAO2P1 11596392 IC50 > 2000 nM T63179 CSB97O 11617028 Ki = 21 nM T63179 CRL3A7 11632925 IC50 = 120 nM T63179 CQB0E3 11633482 IC50 = 65 nM T63179 C9DNG1 11640164 IC50 = 580 nM T63179 C1RJ3I 11646689 IC50 = 1000 nM T63179 CX3L5S 11647533 IC50 = 80 nM T63179 C4S5RG 11655053 IC50 = 175 nM T63179 CDOZ32 11661172 IC50 = 590 nM T63179 C0LEZ3 11667800 Ki = 890 nM T63179 C5XEN0 11668719 IC50 = 220 nM T63179 CZPK72 11682989 IC50 = 80 nM T63179 CCK83U 11690269 IC50 = 160 nM T63179 CY07JH 11696378 IC50 > 2000 nM T63179 CBU02W 11696959 IC50 = 640 nM T63179 C2S9IT 11697271 IC50 = 1900 nM T63179 CGR32I 11697882 IC50 = 340 nM T63179 C75IBX 11704529 IC50 = 90 nM T63179 CGX54N 11704756 IC50 = 210 nM T63179 CO2N1W 11710364 IC50 = 1550 nM T63179 CZ52YQ 11710766 IC50 < 500 nM T63179 C8OPA1 11710962 IC50 = 855 nM T63179 CW3N8H 11711766 IC50 = 280 nM T63179 COEU05 11719039 IC50 = 100 nM T63179 CZ0B7H 11731863 IC50 = 1900 nM T63179 CQO76Z 11741168 IC50 > 2000 nM T63179 C87YNC 11741891 IC50 = 150 nM T63179 CH92VI 11743259 IC50 = 310 nM T63179 C5HLU8 11750204 IC50 = 380 nM T63179 CY1F4I 11752649 Ki = 670 nM T63179 CQU0E7 11774868 IC50 = 435 nM T63179 C4U8KY 12085089 IC50 = 162 nM T63179 C14LTD 15463551 IC50 > 1000 nM T63179 C3QOV0 16099227 IC50 = 430 nM T63179 CW6LO1 16099229 IC50 > 2000 nM T63179 C2R4PK 16099231 IC50 = 450 nM T63179 C9KM7X 16099232 IC50 = 1900 nM T63179 C05CYN 16099234 IC50 = 1600 nM T63179 CJQ8A1 16099236 IC50 = 450 nM T63179 CA72YW 16099237 IC50 > 2000 nM T63179 CS07DB 16099238 IC50 = 98 nM T63179 C42ESN 16099240 IC50 = 580 nM T63179 CMZ91J 16099242 IC50 > 2000 nM T63179 CF69RC 16099243 IC50 > 2000 nM T63179 C60GEM 16099245 IC50 = 1500 nM T63179 CE48CS 16099246 IC50 = 620 nM T63179 CTF2M7 16099247 IC50 = 130 nM T63179 CX9BK2 16099248 IC50 = 775 nM T63179 CN6PA9 16099249 IC50 = 350 nM T63179 C9Z6AK 16099250 IC50 = 120 nM T63179 C5Z8HR 16099251 IC50 = 91 nM T63179 CWK76M 16099252 IC50 = 880 nM T63179 C3BU9M 16216822 IC50 = 290 nM T63179 C1Q5SV 16220168 IC50 = 510 nM T63179 CH6CN0 16658901 Ki > 10000 nM T63179 CU9LS2 16661702 EC50 = 5000 nM T63179 C1UY8J 16666386 IC50 > 1000 nM T63179 CWK35C 16730429 IC50 = 8700 nM T63179 CSKX58 17758233 Ki = 410 nM T63179 C7CPW9 17758234 Ki = 48 nM T63179 CI5KT6 17758236 Ki = 42 nM T63179 C3FP7L 17921933 IC50 = 3162 nM T63179 CX03YG 18188955 IC50 = 1220 nM T63179 CR19ST 18512166 IC50 = 310 nM T63179 CEN14G 18512334 IC50 = 4000 nM T63179 CS9CI5 18551230 IC50 = 30 nM T63179 CBI64N 18551237 IC50 = 130 nM T63179 C5ZYJ0 20231824 Ki = 952 nM T63179 CEH7V5 20786216 IC50 > 1000 nM T63179 C97WCO 21941658 IC50 = 1.259 nM T63179 CCI89R 21948853 IC50 > 1000 nM T63179 CB2SF4 21948904 IC50 > 1000 nM T63179 C2ZP7V 22218142 IC50 = 1500 nM T63179 C1QTK4 22398492 IC50 = 240 nM T63179 C6CSB4 22398502 IC50 > 2000 nM T63179 CR8N1E 22398506 IC50 = 1420 nM T63179 CM83TU 22398533 IC50 = 265 nM T63179 C34LHW 22398559 IC50 = 910 nM T63179 CJBW90 22398592 IC50 > 2000 nM T63179 CEJ65O 22398627 IC50 = 415 nM T63179 CZI4C6 24739672 Ki = 1000 nM T63179 CS23KY 24739834 Ki = 1390 nM T63179 C1M9QG 24739836 Ki = 1770 nM T63179 CG5SJ0 24739997 Ki = 1490 nM T63179 C7Z1HW 24740156 Ki = 1440 nM T63179 CTE1N2 24748569 EC50 > 10000 nM T63179 C4WYE7 24749678 Ki = 1.56 nM T63179 CY2JS4 24749684 Ki = 1.51 nM T63179 C2QHO3 24749808 Ki = 0.319 nM T63179 C5S6JN 24780149 IC50 > 1000 nM T63179 CW5TJ7 24781731 IC50 > 1000 nM T63179 C1JTW2 24851053 Ki = 0.342 nM T63179 CC53XL 24860583 Ki > 3000 nM T63179 C58RHY 24883011 IC50 = 80 nM T63179 CW35CK 24883012 IC50 = 41 nM T63179 C3SC0V 24883054 IC50 = 76 nM T63179 C4SA6C 24883055 IC50 = 15 nM T63179 C5LZK2 24895096 IC50 = 1350 nM T63179 COGP96 24936313 IC50 > 5000 nM T63179 CVY09S 24936449 IC50 > 5000 nM T63179 C06PDG 24952192 EC50 > 5000 nM T63179 CG1CF9 24952193 EC50 > 5000 nM T63179 CZC7L8 24953162 IC50 > 10000 nM T63179 C4W7BN 24954947 IC50 > 10000 nM T63179 C6XC2R 24954951 IC50 > 20000 nM T63179 CYES17 24957737 Ki > 3000 nM T63179 C83YKB 24961057 Ki > 1000 nM T63179 CIGM27 24983460 IC50 = 280 nM T63179 CHY0D7 25013322 IC50 > 10000 nM T63179 C0TPS5 25013653 IC50 > 10000 nM T63179 CWU91M 25013811 IC50 > 10000 nM T63179 CSH29L 25013812 IC50 > 10000 nM T63179 C7QCX0 25052023 IC50 = 2.4 nM T63179 CAW8M0 25070694 IC50 = 2800 nM T63179 C21XDY 25145083 Ki > 10000 nM T63179 CS6JQ1 25167502 Ki = 155 nM T63179 C0XPW9 25168896 IC50 = 340 nM T63179 CUL27D 25168900 IC50 = 260 nM T63179 CEV2D7 25205475 IC50 = 260 nM T63179 C9S0ZW 25205477 IC50 = 330 nM T63179 C49KHR 25206116 IC50 = 510 nM T63179 C9FM2U 42642501 Ki <= 10 nM T63179 CXZ35T 44193145 Ki = 656 nM T63179 C2MOF7 44193146 Ki = 378 nM T63179 CWR6X1 44193147 Ki = 2250 nM T63179 C3JOW4 44193245 Ki = 1470 nM T63179 CHGI03 44251606 IC50 = 475 nM T63179 C0OA6M 44264483 IC50 > 10000 nM T63179 COCE32 44264569 IC50 > 10000 nM T63179 CI0TN2 44264577 IC50 > 10000 nM T63179 CXOR54 44264579 IC50 > 10000 nM T63179 C01HSQ 44264588 IC50 > 10000 nM T63179 CDB54J 44305270 IC50 > 1000 nM T63179 C0XLN6 44305556 IC50 > 1000 nM T63179 C1UK4M 44305720 IC50 = 1889 nM T63179 CH4PU5 44305819 IC50 = 2484 nM T63179 C6N1AR 44305929 IC50 2871 nM T63179 C73CXK 44354006 IC50 = 363 nM T63179 C0N3TD 44354884 IC50 = 2700 nM T63179 CPQ2A6 44354885 IC50 = 1000 nM T63179 CM0G1V 44354886 IC50 = 2000 nM T63179 CL6G3Q 44355066 IC50 = 2100 nM T63179 CSAU31 44377064 IC50 > 10000 nM T63179 C7H9NC 44377081 IC50 > 10000 nM T63179 C60DYH 44377090 IC50 = 2000 nM T63179 CVH2R3 44377098 IC50 = 2900 nM T63179 CYLI63 44377110 IC50 > 10000 nM T63179 CQX39I 44377356 IC50 = 570 nM T63179 C9FJW4 44377382 IC50 = 1900 nM T63179 C13SYV 44396250 Ki = 300 nM T63179 CB1P0S 44396251 Ki = 80 nM T63179 CHY1C3 44396271 Ki = 590 nM T63179 C29MBI 44396272 Ki = 310 nM T63179 C4TQ6N 44396282 Ki = 440 nM T63179 CH2Y3L 44396283 Ki = 190 nM T63179 CWZB52 44396284 Ki = 850 nM T63179 CD80LM 44396296 Ki > 1000 nM T63179 C6SI5L 44396297 Ki > 1000 nM T63179 CR4H1E 44396316 Ki = 510 nM T63179 C45LRH 44396317 Ki = 140 nM T63179 C5JG6H 44396330 Ki > 1000 nM T63179 CA8V4G 44396331 Ki > 1000 nM T63179 C57CPQ 44396332 Ki = 310 nM T63179 CXHF58 44403036 IC50 = 215 nM T63179 C6JNI4 44403038 IC50 = 60 nM T63179 C45SOW 44403039 IC50 = 315 nM T63179 CXZ4S3 44426781 Ki = 3490 nM T63179 C8HO4K 44426782 Ki = 585 nM T63179 C0FEN3 44426790 Ki = 298 nM T63179 C19MJP 44426793 Ki = 527 nM T63179 C1ZDA4 44426795 Ki = 1270 nM T63179 CIOW01 44431179 IC50 = 520 nM T63179 C3SJ5V 44433504 Ki = 7.5 nM T63179 C2SCP7 44435606 IC50 = 1600 nM T63179 CH5E3L 44435611 IC50 > 1300 nM T63179 CDO62N 44435656 IC50 = 650 nM T63179 C9TP4C 44435662 IC50 = 345 nM T63179 C19TMW 44435663 IC50 = 730 nM T63179 C90WUC 44435667 IC50 = 430 nM T63179 CHFB89 44435668 IC50 = 300 nM T63179 C8IWK2 44435669 IC50 = 250 nM T63179 CYG7X4 44473146 IC50 > 10000 nM T63179 CR5SI0 44476535 EC50 > 10000 nM T63179 CM29JD 44516036 IC50 > 10000 nM T63179 CR19IH 44543858 IC50 > 2000 nM T63179 C05HEP 44543860 IC50 > 2000 nM T63179 C45ZHO 44543969 IC50 > 2000 nM T63179 C25OXZ 44544094 IC50 > 2000 nM T63179 C7JIF6 44544321 IC50 > 2000 nM T63179 CF6V4G 44563171 EC50 > 10000 nM T63179 C8BGL6 44585565 IC50 > 3000 nM T63179 CIJP09 44605898 IC50 > 10000000 nM T63179 C9PLK4 45263610 IC50 > 2000 nM T63179 C78JKD 45265930 IC50 = 1100 nM T63179 C08UBE 45272032 IC50 > 10000 nM T63179 C57EZH 45275745 IC50 = 110 nM T63179 CU7D0O 45278780 IC50 = 3.7 nM T63179 CY8A1D 45278857 IC50 = 3.1 nM T63179 CGX87F 45279098 IC50 = 6.5 nM T63179 CL9P2A 45380783 IC50 = 3.8 nM T63179 CKC0B7 46237842 IC50 = 59 nM T63179 C4KN0J 46237981 IC50 = 31 nM T63179 C7KW8T 46883839 EC50 > 10000 nM T63179 CZSG25 46883893 EC50 > 10000 nM T63179 C72MUY 46889765 IC50 > 5000 nM T63179 C6DVO1 46889848 IC50 > 10000 nM T63179 CZ90FC 46894119 Ki = 9 nM T63179 C04KWS 46913888 IC50 = 54 nM T63179 C1U7QL 46913889 IC50 = 52 nM T63179 C3Q7RI 46913890 IC50 = 6 nM T63179 CY7D0I 46913891 IC50 = 80 nM T63179 CQ93ML 46913892 IC50 = 135 nM T63179 C1ZRD2 46914168 IC50 = 1620 nM T63179 CWV42M 46914169 IC50 = 3740 nM T63179 CK6SJ3 46914453 IC50 = 275 nM T63179 C4HQ5Y 46914584 IC50 = 223 nM T63179 C9F4PR 46914585 IC50 = 4340 nM T63179 CZE49A 46914586 IC50 = 553 nM T63179 CGS9U8 46914587 IC50 = 41 nM T63179 C34EDY 46914588 IC50 = 21 nM T63179 CLCI21 46914734 IC50 = 13 nM T63179 C2NM6E 46914737 IC50 = 25 nM T63179 CKP01L 46914738 IC50 = 58 nM T63179 CP91XE 46914741 IC50 = 89 nM T63179 C3Q5PE 46914742 IC50 = 4 nM T63179 C6OG0A 46914743 IC50 = 7 nM T63179 C1TMA8 46914744 IC50 = 150 nM T63179 CE7KZ8 46914881 IC50 = 83 nM T63179 CI0Y4F 46914882 IC50 > 10000 nM T63179 C8HWO7 46914883 IC50 = 784 nM T63179 C6FN4G 46914884 IC50 = 246 nM T63179 CXY74T 46914885 IC50 = 9730 nM T63179 CF1D5Q 46914886 IC50 = 488 nM T63179 CVGF35 46914887 IC50 > 500 nM T63179 C4ZPR6 46915029 IC50 = 180 nM T63179 CXR29C 46915030 IC50 > 10000 nM T63179 C9NC0K 46915031 IC50 = 1440 nM T63179 CY3O2C 46915043 IC50 = 41 nM T63179 CHG94E 46915044 IC50 = 32 nM T63179 CK85FJ 46915045 IC50 = 101 nM T63179 CQ6J3N 46915201 IC50 = 2080 nM T63179 CC84WO 46915202 IC50 = 8360 nM T63179 CTM2J5 46915203 IC50 = 31 nM T63179 C75IFZ 46915353 IC50 = 16 nM T63179 CJW51A 46915354 IC50 = 26 nM T63179 CX70GY 46915355 IC50 = 15.2 nM T63179 CPTL45 46915356 IC50 = 2 nM T63179 C39SUV 46915640 IC50 = 243 nM T63179 CX6WK5 46915641 IC50 = 535 nM T63179 CW8J2E 46915642 IC50 = 56 nM T63179 C05YTF 46915643 IC50 = 284 nM T63179 CMW7E4 46915644 IC50 = 56 nM T63179 CA43UG 46915645 IC50 > 127 nM T63179 CJ3DN2 46915781 IC50 > 1000 nM T63179 C4L1JF 46915782 IC50 = 383 nM T63179 CB4X3D 46915783 IC50 > 10000 nM T63179 CK7DI0 46915784 IC50 > 10000 nM T63179 CU7L4T 46915785 IC50 = 10000 nM T63179 CE9OU3 46915786 IC50 = 410 nM T63179 CI3E2M 46915787 IC50 = 763 nM T63179 C1BV5K 46916070 IC50 = 3650 nM T63179 C06JHQ 46916071 IC50 = 441 nM T63179 CQ37UY 46916072 IC50 = 1590 nM T63179 C38HIP 46916073 IC50 = 1290 nM T63179 CPK95L 46916074 IC50 = 151 nM T63179 C7NC4B 46917090 IC50 = 2.8 nM T63179 C2LCJ7 46937290 IC50 = 210 nM T63179 CKQ8J3 46937431 IC50 > 2000 nM T63179 CL7P3N 46938234 IC50 = 1.8 nM T63179 COS28G 46938235 IC50 = 18 nM T63179 CFJT93 46938236 IC50 = 7.6 nM T63179 CHL70M 46938239 IC50 = 4.1 nM T63179 C8P7JH 46938914 IC50 > 2000 nM T63179 CY95VK 46938915 IC50 > 2000 nM T63179 CVX25Q 46938916 IC50 = 220 nM T63179 C2V5AT 46939019 IC50 = 480 nM T63179 C5R6GI 46939020 IC50 = 390 nM T63179 CF1BX0 46939115 IC50 > 2000 nM T63179 C4P0EU 46939116 IC50 = 160 nM T63179 CD6B7X 46939395 IC50 = 58 nM T63179 C1KXF2 46939396 IC50 > 2000 nM T63179 CVN4W1 47958757 IC50 = 168 nM T63179 CX0NO8 49782554 EC50 < 15848.93 nM T63179 CC7T8Q 49782555 EC50 < 15848.93 nM T63179 CD07EV 49782777 EC50 < 15848.93 nM T63179 C43UKW 49782778 IC50 < 14421.15 nM T63179 C2JTF0 49782779 EC50 < 15848.93 nM T63179 CS7KX9 49782780 IC50 < 12560.3 nM T63179 C36RYU 49782781 IC50 = 5140.44 nM T63179 C8OA0C 49782985 EC50 < 15848.93 nM T63179 C5Y6QU 49782986 EC50 < 15848.93 nM T63179 CB8V7R 49782987 EC50 < 15848.93 nM T63179 CU3S6H 49836028 EC50 > 5000 nM T63179 C96SLW 49851364 EC50 > 5000 nM T63179 CDN4K6 49851369 EC50 > 5000 nM T63179 C4YXN1 49851467 EC50 > 5000 nM T63179 CUD91T 49862248 EC50 > 10000 nM T63179 C5NX4D 49864061 IC50 = 2530 nM T63179 CPH9D8 49864098 IC50 = 69 nM T63179 CMS1N3 49864127 IC50 = 15 nM T63179 CTE0N7 49864128 IC50 = 720 nM T63179 COP7W2 49864129 IC50 = 127 nM T63179 CCKJ45 49864153 IC50 = 849 nM T63179 C19FRV 49864154 IC50 = 65 nM T63179 CWGD27 49864174 IC50 = 146 nM T63179 C9YCN1 49864175 IC50 = 39 nM T63179 CTKV39 49864176 IC50 = 26 nM T63179 CZ8J1V 50942115 Ki = 800 nM T63179 C23OEF 50942312 EC50 > 10000 nM T63179 CX1KO8 51346768 Ki = 849 nM T63179 C7N9TD 51346823 Ki = 1518 nM T63179 C0WDX3 51347001 Ki = 1115 nM T63179 CF8DK7 51347002 Ki = 3170 nM T63179 CTH45Q 52918523 IC50 > 10000 nM T63179 CL8D1Z 52921432 IC50 = 130 nM T63179 CEC4I7 52941608 IC50 = 230 nM T63179 CDV90J 52942528 IC50 > 1000 nM T63179 C8Y9SU 52944898 IC50 > 1000 nM T63179 CK5UT4 53317489 Ki = 126 nM T63179 CM0LU1 53318659 Ki = 1200 nM T63179 CUD48O 53320087 Ki = 0.64 nM T63179 CD0N1K 53323476 IC50 = 356 nM T63179 CYH3V0 53325642 Ki = 86.8 nM T63179 C82DYI 53326614 Ki > 4170 nM T63179 CJCP75 53359074 EC50 > 5000 nM T63179 C9H5YE 53361128 EC50 > 5000 nM T63179 CUR24K 53875787 IC50 = 2800 nM T63179 C1JR5W 54576068 IC50 = 24 nM T63179 CS62XZ 54590901 IC50 = 53.9 nM T63179 C30XLO 54592009 Ki = 6.3 nM T63179 CCS8R6 54592010 IC50 = 39 nM T63179 CML2E7 54592011 IC50 = 86 nM T63179 CRVB01 54592087 IC50 = 266 nM T63179 C7W1BA 54592088 IC50 = 109 nM T63179 C9N3IS 54592089 IC50 = 56 nM T63179 C2GML6 54592090 IC50 = 33 nM T63179 C05FVP 54592092 IC50 = 19 nM T63179 C9W5DZ 56593984 EC50 > 5000 nM T63179 CF3G2M 56925477 IC50 = 36 nM T63179 CZ7O8G 56925478 IC50 = 69 nM T63179 CV5C0T 56925479 IC50 > 10000 nM T63179 C9ITY0 56925480 IC50 > 10000 nM T63179 C3M4TE 56925570 IC50 = 920 nM T63179 CZ4I2J 56925571 IC50 = 6800 nM T63179 CW87RG 56925573 IC50 = 2000 nM T63179 C4Z5LF 56925574 IC50 = 4100 nM T63179 CKF8Z3 56925575 IC50 = 1300 nM T63179 CY20OR 56925668 IC50 > 10000 nM T63179 C30DAL 56925669 IC50 = 600 nM T63179 CQHA65 56925670 IC50 = 310 nM T63179 CJP31U 56925671 IC50 = 270 nM T63179 CV86DS 56925673 IC50 = 2700 nM T63179 CI3S6F 56925790 IC50 = 5300 nM T63179 CTY1Q9 56925791 IC50 = 1100 nM T63179 CH40YG 56925792 IC50 = 960 nM T63179 C2PLD4 56925793 IC50 = 260 nM T63179 CU02HT 56925794 IC50 = 570 nM T63179 CM19WI 56925904 IC50 > 10000 nM T63179 CA7BX4 56925905 IC50 = 440 nM T63179 CTR7X3 56925906 IC50 = 1100 nM T63179 C39VBK 56925907 IC50 = 430 nM T63179 CV7EN5 56925908 IC50 = 320 nM T63179 CU69SK 56925909 IC50 = 590 nM T63179 CAMI87 56925910 IC50 = 700 nM T63179 CTG9I7 56926011 IC50 = 70 nM T63179 CPD82H 56968080 IC50 = 7.1 nM T63179 CM0SG2 57390990 IC50 = 1100 nM T63179 CU8AN3 57392780 IC50 = 790 nM T63179 CX12JM 57392781 IC50 = 45 nM T63179 C9OMW1 57392782 IC50 = 405 nM T63179 C30JOV 57394501 IC50 = 190 nM T63179 CINU04 57396254 IC50 = 225 nM T63179 C1O6JU 57396255 IC50 = 230 nM T63179 CVOB64 57399718 IC50 = 610 nM T63179 CF83VM 57401459 EC50 > 5000 nM T63179 C7W3YD 57401479 IC50 = 430 nM T63179 CR6L7E 57403222 IC50 = 1450 nM T63179 CPU6W7 57473898 IC50 = 80 nM T63179 CEJ25K 57473899 IC50 = 270 nM T63179 CUJ08D 57474008 IC50 = 70 nM T63179 CDB0F1 57503322 IC50 = 39 nM T63179 CIDS61 57503325 IC50 = 19 nM T63179 C2U1GQ 57524309 IC50 = 22 nM T63179 C0BDS9 57585514 IC50 < 2 nM T63179 CM17UZ 57585515 IC50 = 47 nM T63179 CYGU85 57585534 IC50 = 1.3 nM T63179 C3WG0L 57666312 Ki = 1100 nM T63179 C43GDR 57666397 Ki = 290 nM T63179 CTM6K5 57690900 IC50 > 5000 nM T63179 CB2I7A 57748722 Ki <= 10 nM T63179 CT9Y6X 57748723 Ki <= 10 nM T63179 C6J0HD 57748748 Ki <= 10 nM T63179 C2MFH6 57748755 Ki <= 10 nM T63179 CMR56T 57748765 Ki <= 10 nM T63179 C05UIP 57748768 Ki <= 10 nM T63179 CH2PV6 57748780 Ki = 0.79 nM T63179 CL13HZ 57748781 Ki = 0.4 nM T63179 C7UH3N 57748789 Ki <= 10 nM T63179 C2YT7S 57748790 Ki = 0.23 nM T63179 C1KZT3 57906156 IC50 = 500 nM T63179 C3IN9F 57983276 IC50 = 170 nM T63179 CJ6Y1B 58026134 IC50 > 2000 nM T63179 C19XQV 58026164 IC50 > 2000 nM T63179 CR7H3O 58026170 IC50 > 2000 nM T63179 C7XL3D 58026176 IC50 > 2000 nM T63179 CT1EM3 58064710 IC50 = 3.7 nM T63179 C8S3EQ 58064714 IC50 = 2.7 nM T63179 CPI62D 58064720 IC50 = 2.2 nM T63179 CL42XF 58064726 IC50 = 4.3 nM T63179 CPL9A6 58064729 IC50 = 55.9 nM T63179 CRFS78 58064730 IC50 = 3.3 nM T63179 CN1J3V 58064734 IC50 = 17.8 nM T63179 CA0SH5 58064735 IC50 = 4.4 nM T63179 CI7BP4 58064741 IC50 = 21.4 nM T63179 C2FZA7 58064756 IC50 = 9.4 nM T63179 C3AMO0 58064757 IC50 = 4450 nM T63179 C47AUR 58392644 EC50 = 2.5 nM T63179 C9CQS0 58392665 EC50 = 3.2 nM T63179 CXF39M 58392685 EC50 > 3000 nM T63179 C7FXH3 58392721 EC50 > 3000 nM T63179 CJDN90 58392790 EC50 = 1.6 nM T63179 CO59DQ 58392803 EC50 > 3000 nM T63179 C5K9PJ 58483018 IC50 = 1.2 nM T63179 C4C2FT 58599563 IC50 = 1300 nM T63179 CWAD17 58731166 Ki <= 500 nM T63179 CNE02T 58731180 Ki <= 500 nM T63179 CVS58C 58731199 Ki <= 500 nM T63179 C3VU0Q 58731202 Ki <= 500 nM T63179 C03HFM 58731234 Ki <= 500 nM T63179 CADQ18 58731243 Ki <= 500 nM T63179 CI7XQ5 58731245 Ki <= 500 nM T63179 C67UET 58731323 Ki <= 500 nM T63179 C0JL7A 58973277 IC50 > 1000 nM T63179 CY38HG 59233337 Ki > 1000 nM T63179 CUX4E7 59233347 Ki > 3333 nM T63179 CO63VJ 59233364 Ki > 1000 nM T63179 C2A9JO 59251119 IC50 > 5000 nM T63179 CD8A6P 59281281 IC50 = 49 nM T63179 CBZ0M5 59281312 IC50 = 170 nM T63179 CCT59B 59281329 IC50 = 510 nM T63179 CQI5C4 59281343 IC50 = 38 nM T63179 CH5E1F 59281346 IC50 > 10000 nM T63179 CPE83R 59281354 IC50 = 180 nM T63179 CI9EP1 59281363 IC50 = 8.4 nM T63179 CQ2BO1 59281403 IC50 = 51 nM T63179 CP78RD 59281411 IC50 = 95 nM T63179 CCNU12 59281412 IC50 = 10 nM T63179 C7HVB1 59281416 IC50 = 490 nM T63179 CE5A0V 59281447 IC50 = 75 nM T63179 CZT9S6 59281449 IC50 = 430 nM T63179 CIKQ89 59281508 IC50 = 990 nM T63179 CE1A7J 59281531 IC50 = 680 nM T63179 CK9JZ4 59281538 IC50 = 36 nM T63179 C4TG5U 59281540 IC50 = 22 nM T63179 CPC80S 59281541 IC50 = 64 nM T63179 CXS5C4 59281543 IC50 = 250 nM T63179 C7KPR9 59281566 IC50 = 150 nM T63179 CUJP64 59281599 IC50 = 600 nM T63179 CYZI85 59556974 IC50 > 10000 nM T63179 C5C3AO 59770003 Ki = 2.48 nM T63179 CH36PL 59807625 IC50 < 500 nM T63179 C54ATL 59807726 IC50 < 500 nM T63179 C8S7OB 59808080 IC50 < 500 nM T63179 CYU57B 59808129 IC50 < 500 nM T63179 C2TNO8 60026286 IC50 > 2000 nM T63179 CZE5J8 60026377 IC50 > 2000 nM T63179 C0LDS2 60026592 IC50 = 1150 nM T63179 C31PTC 60026641 IC50 > 2000 nM T63179 C67NSE 60026675 IC50 > 2000 nM T63179 C6GP5R 60026731 IC50 = 720 nM T63179 C5M8HV 60026772 IC50 = 1200 nM T63179 CI36XS 60026787 IC50 > 2000 nM T63179 C3JD8M 60026802 IC50 > 2000 nM T63179 CE9MI4 60026817 IC50 = 1900 nM T63179 C04EKW 60026878 IC50 > 2000 nM T63179 CPRW14 66991384 IC50 = 160 nM T63179 CYP31Z 66995780 IC50 = 3050 nM T63179 CK36QI 66996020 IC50 > 10000 nM T63179 CJ09TZ 66996063 IC50 = 2225 nM T63179 C3EU7N 66996137 IC50 = 276 nM T63179 C1CXY9 66996546 IC50 = 401 nM T63179 C9Y2DN 66996560 IC50 = 727 nM T63179 C9LOZ1 66996568 IC50 = 1181 nM T63179 CH39DP 67053383 IC50 > 2000 nM T63179 C3LF8O 67053425 IC50 > 2000 nM T63179 CMYP75 67415874 IC50 = 100 nM T63179 CQU8E3 68031408 IC50 = 11 nM T63179 C1FK3D 69081573 IC50 = 31 nM T63179 CB6HX8 69082589 IC50 = 480 nM T63179 C43PON 69675755 IC50 = 9.4 nM T63179 COR52G 69675880 IC50 = 13 nM T63179 C9Q7VH 70561849 IC50 = 39 nM T63179 CARO49 70685018 Ki = 150 nM T63179 C5QPC0 70697572 Ki = 170 nM T63179 C94FCP 71452686 IC50 = 3000 nM T63179 CF08ME 71457470 Ki = 0.4 nM T63179 CEO5G4 71461616 IC50 = 1900 nM T63179 C78IOK 71467161 IC50 = 310 nM T63179 C1MHC0 71467246 IC50 = 47 nM T63179 C4B0IC 71467248 IC50 = 26 nM T63179 CYW34A 71519686 IC50 = 120 nM T63179 CGK4S8 71543393 Ki = 1450 nM T63179 C83YJF 71544946 IC50 = 39 nM T63179 CK2O1Z 71545110 IC50 = 54 nM T63179 C0LD8K 71548690 IC50 = 270 nM T63179 C19CGP 71548691 IC50 = 1700 nM T63179 C4BE6G 71548692 IC50 = 1110 nM T63179 CCK7Q3 71548693 IC50 = 240 nM T63179 CK9S0J 71548694 IC50 = 1440 nM T63179 CT9Y5D 71549558 Ki = 2 nM T63179 C8ZX0F 71549573 IC50 = 180 nM T63179 COQ5C4 71549690 IC50 = 230 nM T63179 CE7NZ0 71549691 IC50 = 190 nM T63179 C1ZF5V 71549692 IC50 = 180 nM T63179 C15JLF 71549694 IC50 = 120 nM T63179 CUX57Y 71549702 IC50 = 200 nM T63179 CQX42S 71549703 IC50 = 190 nM T63179 CZ3C8X 71549705 IC50 = 500 nM T63179 C0IH6J 71549706 IC50 = 170 nM T63179 CZ8Y7O 71549829 IC50 = 40 nM T63179 CPS61I 71549840 IC50 = 37 nM T63179 CC5AU3 71549841 IC50 = 55 nM T63179 CCV90M 71549842 IC50 = 14 nM T63179 CPFL57 71549843 IC50 = 33 nM T63179 CY8SP0 71549969 IC50 = 210 nM T63179 CXP57U 71549980 IC50 = 180 nM T63179 CA64KN 71550109 IC50 = 400 nM T63179 CUG9C6 71550110 IC50 = 30 nM T63179 CK7NS4 71550116 IC50 = 270 nM T63179 COW8K4 71550118 IC50 = 340 nM T63179 C50TXO 71550241 IC50 = 33 nM T63179 CX6JR5 71550242 IC50 = 34 nM T63179 C93KZM 71550243 IC50 = 42 nM T63179 C6WIA2 71550244 IC50 = 120 nM T63179 CX26UJ 71550250 IC50 = 990 nM T63179 C7R1LJ 71550386 IC50 = 800 nM T63179 CMVD92 71550387 IC50 = 150 nM T63179 CUK7A8 71550511 IC50 = 160 nM T63179 CYB2L0 71550527 IC50 = 230 nM T63179 C6XF9J 71550528 IC50 = 370 nM T63179 CJYQ15 71550529 IC50 = 170 nM T63179 CSHT69 71550657 IC50 = 82 nM T63179 CJX19L 71550659 IC50 = 1530 nM T63179 C6SNW1 71550660 IC50 = 130 nM T63179 CU0Q9P 71550799 IC50 = 470 nM T63179 C8SDX6 71550801 IC50 = 68 nM T63179 CK3HZ0 71550802 IC50 = 240 nM T63179 C9QD8V 71726436 IC50 = 300 nM T63179 CKO01U 71726437 IC50 > 40000 nM T63179 CP9M2C 71726438 IC50 = 750 nM T63179 C6TXD3 71726439 IC50 = 450 nM T63179 CP62QW 71726440 IC50 > 40000 nM T63179 CQYH84 71726556 IC50 > 40000 nM T63179 C8N4UF 71726557 IC50 > 40000 nM T63179 C6TXF5 71726558 IC50 = 500 nM T63179 C4RY0L 71726559 IC50 = 400 nM T63179 CPL35F 71726560 IC50 = 2900 nM T63179 C07YPM 71726687 IC50 > 40000 nM T63179 C6OQT5 71726688 IC50 > 40000 nM T63179 C7F3PL 71726689 IC50 > 40000 nM T63179 C91RTU 71726690 IC50 > 40000 nM T63179 CAR9T3 71726691 IC50 > 40000 nM T63179 C1E3QT 71726810 IC50 > 10000 nM T63179 CV02SB 71726811 IC50 > 40000 nM T63179 C0OXK4 71726812 IC50 > 40000 nM T63179 CL8Z2I 71726813 IC50 = 250 nM T63179 CWS86Q 71726934 IC50 = 3000 nM T63179 C62XFJ 71726935 IC50 > 10000 nM T63179 CIR49D 71726936 IC50 > 40000 nM T63179 CMO7T2 71726937 IC50 = 13000 nM T63179 CE67IF 71726938 IC50 = 16000 nM T63179 CEI4R9 71726939 IC50 > 40000 nM T63179 CKFV04 71727059 IC50 = 2500 nM T63179 CEK6Y8 71727060 IC50 = 1500 nM T63179 CJ0Z6D 71727061 IC50 = 3000 nM T63179 CAG0M9 71727062 IC50 = 300 nM T63179 CN4TI1 71727063 IC50 = 4000 nM T63179 CB45XH 71727183 IC50 = 15000 nM T63179 C76QBF 71727184 IC50 > 40000 nM T63179 CIY4W8 71727185 IC50 > 40000 nM T63179 CB12CL 71727731 IC50 = 6000 nM T63179 C91POE 71727732 IC50 = 1000 nM T63179 C6O2YB 71727733 IC50 = 300 nM T63179 CIUT23 71727734 IC50 = 1000 nM T63179 CE6GH7 71727735 IC50 = 500 nM T63179 CDME45 71727852 IC50 = 3000 nM T63179 C8W7UV 71727853 IC50 = 200 nM T63179 CLTX21 71727854 IC50 = 280 nM T63179 CG0Y6I 71727855 IC50 = 400 nM T63179 C6A1KB 71727856 IC50 = 2600 nM T63179 CRS9A7 71727980 IC50 = 570 nM T63179 CRC7E9 71727981 IC50 = 500 nM T63179 CCK75S 71727982 IC50 > 10000 nM T63179 C3X0QV 71727983 IC50 = 3000 nM T63179 C2KIM1 71727984 IC50 = 600 nM T63179 CKQN54 71728108 IC50 = 2000 nM T63179 C2W9HE 71728109 IC50 = 1000 nM T63179 CVL7Q6 71728110 IC50 = 100 nM T63179 CM78AL 71728111 IC50 = 300 nM T63179 CN80TQ 71728112 IC50 = 100 nM T63179 CF52OE 71728113 IC50 = 4000 nM T63179 C8BGF3 71728224 IC50 = 1200 nM T63179 CJ4M6P 71728225 IC50 = 2000 nM T63179 C10AOX 71728227 IC50 > 30000 nM T63179 C4XSM7 71728228 IC50 = 3000 nM T63179 CW5C6N 71728229 IC50 = 280 nM T63179 CP5KM8 72163477 IC50 = 660 nM T63179 CA6O4K 72163478 IC50 = 750 nM T63179 C27XWS 72163479 IC50 = 1200 nM T63179 C6M9CN 72163480 IC50 = 120 nM T63179 CL8AH4 72163481 IC50 = 550 nM T63179 CB2SD9 72163621 IC50 = 1200 nM T63179 CU6NA8 72163622 IC50 = 170 nM T63179 CTEV75 72163623 IC50 = 33 nM T63179 CER73F 72163624 IC50 = 68 nM T63179 CC8VM7 72163625 IC50 = 1600 nM T63179 CS69AC 72163626 IC50 = 94 nM T63179 CAJ0H5 72163627 IC50 = 43 nM T63179 C1D3EU 72163754 IC50 = 92 nM T63179 C1G3ES 72163755 IC50 = 23 nM T63179 CP8AC2 72188914 EC50 > 5000000 nM T63179 CA6FO5 72188915 EC50 > 5000000 nM T63179 CZ5O6M 72204151 IC50 = 3500 nM T63179 CGT02E 72204156 IC50 = 10900 nM T63179 CW6I9L 72204538 EC50 = 4100 nM T63179 CH5Q8D 72544150 IC50 = 40 nM T63179 C4YUD1 72544151 IC50 = 45 nM T63179 CTM6Y0 72544152 IC50 = 2029 nM T63179 C2K7JR 72544153 IC50 = 1393 nM T63179 C0ZGC8 72544374 IC50 = 1530 nM T63179 CC64LQ 72544375 IC50 = 1974 nM T63179 CNG1C6 72544376 IC50 = 4698 nM T63179 CS1QT2 72544377 IC50 = 121 nM T63179 C0X6YV 72544378 IC50 = 1207 nM T63179 C97CRH 72544379 IC50 = 342 nM T63179 CJ8N2H 72544380 IC50 = 1844 nM T63179 CRB36F 72544601 IC50 = 2086 nM T63179 C3LJ6V 72544602 IC50 = 627 nM T63179 C34FBN 72544603 Ki = 113 nM T63179 CLA3Y9 72710581 Ki = 6.1 nM T63179 CXB45U 72724690 IC50 = 270 nM T63179 CI2K6C 72725442 IC50 = 700 nM T63179 C0W2UD 72725443 IC50 = 400 nM T63179 CQ5D1B 72725444 IC50 = 1100 nM T63179 C2PJV7 72725445 IC50 > 10000 nM T63179 CQ4Z2C 72725446 IC50 = 350 nM T63179 C47IMQ 72725447 IC50 = 2400 nM T63179 CJSK52 72725491 IC50 = 360 nM T63179 CS6J4T 72725492 IC50 = 400 nM T63179 C41FYD 72725493 IC50 = 150 nM T63179 CUG96L 72725494 IC50 = 190 nM T63179 CFHJ16 72725495 IC50 = 400 nM T63179 CW7IY3 72725496 IC50 = 330 nM T63179 CSV1I7 72725497 IC50 = 240 nM T63179 COV09R 72725548 IC50 = 320 nM T63179 CTE01I 72725549 IC50 = 1400 nM T63179 C09ZFS 72725550 IC50 = 480 nM T63179 C2Z7QT 72725551 IC50 = 110 nM T63179 C0K2CP 72725552 IC50 = 5200 nM T63179 C37MEN 72725553 IC50 = 1000 nM T63179 CYSM01 72725554 IC50 = 2300 nM T63179 COU49R 76314656 IC50 = 170 nM T63179 C95NBT 76314657 IC50 > 2000 nM T63179 CL95NP 76317025 IC50 = 609 nM T63179 CZ08OF 76317198 IC50 = 510 nM T63179 CR5B2V 76317199 IC50 = 470 nM T63179 C5YFZ6 76318225 IC50 > 2000 nM T63179 C0RK5D 76321918 IC50 = 1100 nM T63179 C3IC5B 76329113 IC50 > 2000 nM T63179 C1RB6X 76329114 IC50 = 260 nM T63179 CP8M1Z 76332766 IC50 > 2000 nM T63179 CKDI18 76332767 IC50 > 2000 nM T63179 CK21EY 77461202 IC50 = 420 nM T63179 CX20VN 84429708 Ki = 1000 nM T63179 CIU65X 86280440 Ki = 1580 nM T63179 CH46CP 87361539 Ki = 0.08 nM T63179 CT50AL 87539277 IC50 > 1000 nM T63179 CY05IC 87733533 IC50 > 1000 nM T63179 C9EH7I 89500376 Ki > 7010 nM T63179 C0EQS7 89501406 Ki = 415 nM T63179 CG67BU 89508836 IC50 = 130 nM T63179 CBLU18 89509944 IC50 = 380 nM T63179 C8JG7O 89510193 Ki = 1840 nM T63179 CK5D1A 90395281 IC50 = 220 nM T63179 CPC47K 90396922 IC50 = 1600 nM T63179 CQ06RH 90654508 IC50 = 1300 nM T63179 CY5L7N 90655674 IC50 = 660 nM T63179 C9B0QF 90655675 IC50 = 1320 nM T63179 CG6QP2 90655676 IC50 = 670 nM T63179 C8EH0K 90655677 IC50 = 6740 nM T63179 C8GQ4S 90655678 IC50 = 270 nM T63179 C6VZ7X 90656360 IC50 = 9 nM T63179 CNCB43 90656361 IC50 = 10.7 nM T63179 CS42NY 90656362 IC50 = 30.7 nM T63179 C2ZF7W 110763791 Ki = 630.96 nM T63179 CD7RS9 118599615 Ki = 3.981 nM T63179 C70AOV 118599714 Ki = 63.1 nM T63179 C8XLO9 118599727 EC50 = 12.59 nM T63179 CYCM67 118599740 IC50 > 10000 nM T63179 CW7G4T 118599742 Ki = 2.512 nM T63179 C9L5EW 118599756 Ki = 158.49 nM T63179 CVIW94 118599769 EC50 = 1 nM T63179 CFS28Y 118599779 Ki = 50.12 nM T63179 CLS7C1 118707978 EC50 > 5000 nM T63179 C9LV0M 118707979 EC50 > 5000 nM T63179 CC2H4E 118714881 IC50 = 710 nM T63179 C2MQ3P 118714882 IC50 > 10000 nM T63179 CE3I9T 118723172 IC50 > 2000 nM T63179 C13AIC 118723173 IC50 > 2000 nM T63179 C21SWI 118723174 IC50 > 2000 nM T63179 CKR24J 118723175 IC50 > 2000 nM T63179 C28YZF 118723176 IC50 > 2000 nM T63179 C6AGI7 118723177 IC50 > 2000 nM T63179 C4QO8E 118723178 IC50 > 2000 nM T63179 C1RYW9 118796369 Ki = 2 nM T63179 C0X8SA 122178358 IC50 = 1200 nM T63179 C14KFA 122178359 IC50 = 420 nM T63179 C04DIU 122178360 IC50 = 62 nM T63179 CG13LX 122178361 IC50 = 39 nM T63179 C40DRP 122178362 IC50 = 120 nM T63179 C6IV5P 122178363 IC50 = 36 nM T63179 C3MLD0 122178364 IC50 = 64 nM T63179 C0NEZ7 122178365 IC50 = 72 nM T63179 CIT71M 122178366 IC50 = 150 nM T63179 C5ON0U 122178367 IC50 = 1100 nM T63179 C9LIR4 122179356 Ki = 337 nM T63179 CUI57B 122179357 Ki > 3000 nM T63179 CY18QG 122186737 Ki = 2120 nM T63179 C0OR2H 122186738 Ki = 6530 nM T63179 CU0Y8B 122186739 Ki = 3890 nM T63179 CWF0Q4 122186740 Ki = 38.4 nM T63179 CBE6Q8 122186741 Ki = 3880 nM T63179 CX13DR 122186742 Ki = 4250 nM T63179 CJ74HX 122186743 Ki = 3920 nM T63179 C05VWL 122186744 Ki = 44.7 nM T63179 CNX5H4 122186745 Ki = 4470 nM T63179 CQ6BG8 122186747 Ki = 2.1 nM T63179 CH8O2M 122186748 Ki = 27.4 nM T63179 C4LRN1 122186749 Ki = 225 nM T63179 CCK36V 127029882 Ki = 6 nM T63179 CVC84H 127029883 Ki = 6 nM T63179 CFY1P0 127029884 Ki = 6 nM T63179 CU1S6C 127029885 Ki = 7 nM T63179 CA1J0H 127030193 Ki = 1080 nM T63179 CU8Y7N 127030224 Ki = 31 nM T63179 CTEA14 127030225 IC50 = 56 nM T63179 CQ74CG 127030810 Ki = 162 nM T63179 CS5JP0 127031149 Ki = 694 nM T63179 CBW17G 127031150 Ki = 13 nM T63179 C19DUV 127031151 Ki = 14 nM T63179 CLDC46 127031152 Ki = 19 nM T63179 C60SMC 127031153 Ki = 16 nM T63179 C21UAK 127032030 Ki = 144 nM T63179 CBT43F 127032031 Ki = 258 nM T63179 C8TG9C 127032032 Ki = 980 nM T63179 CKZ3X7 127032033 Ki = 55 nM T63179 C8SOU3 127032034 Ki = 230 nM T63179 C87NBI 127032035 Ki = 1452 nM T63179 CKA18M 127032339 Ki > 10 nM T63179 CBR31K 127033260 Ki = 20 nM T63179 CAN7K2 127034410 IC50 = 5217 nM T63179 CSC7I2 127034411 Ki = 1092 nM T63179 C9TG2N 134137487 IC50 > 1000 nM T63179 CTF0J3 135567449 Ki = 1.995 nM T63179 CN24YZ 135567451 EC50 = 0.05012 nM T63179 CPF3B4 135567452 Ki = 0.631 nM T63179 C5MXO2 136000568 Ki > 10000 nM T63179 CM6OX5 136000656 Ki = 2700 nM T63179 CZ2D6U 136059148 Ki = 1600 nM T63179 C6HOU3 136059149 Ki = 1040 nM T63179 CE1G9O 136059150 Ki = 1700 nM T63179 C7LSN6 136088946 Ki = 2800 nM T63179 C3SE8T 136216705 IC50 = 700 nM T63179 CZXM35 136216706 IC50 = 900 nM T63179 CX8H9R 137632028 IC50 = 3900 nM T63179 C0XZC3 137633972 IC50 = 1400 nM T63179 COI80Z 137634236 IC50 > 1000 nM T63179 CP2C7M 137635745 IC50 = 55 nM T63179 CPD87Y 137639726 IC50 > 1000 nM T63179 C3K6DU 137640356 IC50 = 4600 nM T63179 CHTB16 137642739 IC50 = 900 nM T63179 C7KIR1 137643684 IC50 = 6.2 nM T63179 C0J8FI 137646168 IC50 = 4800 nM T63179 CPNB08 137646648 Ki = 195.7 nM T63179 C30ZJF 137648477 IC50 > 1000 nM T63179 C7IG3B 137649694 IC50 = 25 nM T63179 CX63RY 137650280 IC50 = 900 nM T63179 CXWF54 137652695 IC50 = 1100 nM T63179 C69ECN 137653076 IC50 = 18 nM T63179 C8OP2T 137653676 IC50 = 2200 nM T63179 CO92KL 137654415 IC50 > 1000 nM T63179 C8PR9K 137654628 IC50 = 33.4 nM T63179 CX65AR 137656053 IC50 = 1400 nM T63179 CS29XF 137656107 Ki <= 10 nM T63179 C0PL8V 137658165 IC50 = 7 nM T63179 C9GQB2 137658303 IC50 = 1600 nM T63179 C5T7IK 147930449 Ki = 3.981 nM T63179 CCDV87 155511242 IC50 = 114 nM T63179 C28RHM 155514304 Ki = 125.89 nM T63179 CE2YJ9 155514399 Ki = 10 nM T63179 CQF09V 155516050 Ki = 50.12 nM T63179 CQ2GH0 155517818 IC50 = 6309.57 nM T63179 CELU49 155517819 IC50 > 10000 nM T63179 C2E4XV 155518137 Ki = 1000 nM T63179 C4QAB0 155518139 Ki = 1258.93 nM T63179 CCO0Z4 155519877 Ki = 10 nM T63179 C8BD6Y 155522508 Ki = 12.59 nM T63179 CILC13 155524288 IC50 = 5940 nM T63179 C71VIK 155525344 EC50 = 12.59 nM T63179 C1WAQ6 155527406 Ki = 199.53 nM T63179 C5T2QN 155528866 IC50 = 100 nM T63179 CBO7E4 155528935 Ki = 501.19 nM T63179 CQM89D 155529443 Ki < 0.3162 nM T63179 CR0N3F 155529454 Ki = 7.943 nM T63179 CB0XS4 155529625 IC50 > 10000 nM T63179 CLC65H 155532000 Ki = 1995.26 nM T63179 C3HFZ6 155534085 IC50 > 10000 nM T63179 CF52DM 155535034 Ki = 0.5012 nM T63179 CXR2W1 155536089 IC50 = 22 nM T63179 C3FON4 155537084 Ki = 398.11 nM T63179 CUI53F 155537601 Ki = 794.33 nM T63179 C78ISM 155540009 IC50 = 567 nM T63179 CIAW80 155544156 IC50 = 21990 nM T63179 C76OVS 155544396 Ki = 1000 nM T63179 CR6UY8 155545121 IC50 = 20 nM T63179 CE3VY8 155550102 Ki = 6309.57 nM T63179 C6H2ML 155552723 Ki = 7.943 nM T63179 CW8BH4 155554673 Ki = 39.81 nM T63179 C9WV3L 155556878 Ki = 15.85 nM T63179 CR5ZI2 155557239 IC50 = 63.1 nM T63179 CPY83L 155558503 IC50 > 10000 nM T63179 CFAN82 155561077 Ki = 63.1 nM T63179 CQ7HG2 155561626 Ki = 3.162 nM T63179 CXQ23E 155562099 IC50 = 7690 nM T63179 CD4K6Z 155564467 Ki = 0.3162 nM T63179 CS25QB 155564604 IC50 = 32 nM T63179 C7YK6N 155565026 IC50 = 64 nM T63179 C4XJU2 155565054 Ki = 501.19 nM T63179 CPX2J5 155566857 Ki > 6309.57 nM T63179 C79WFJ 155567245 IC50 > 10000 nM T63179 CME1B7 155567676 Ki = 316.23 nM T63179 D00ZGW 46883841 EC50 > 10000 nM T63179 D01ETZ 261000 Ki = 0.54 nM T63179 D01NVD 46830196 EC50 > 19952.62 nM T63179 D04UDT 10407950 IC50 = 126 nM T63179 D07KWO 9823099 IC50 = 6300 nM T63179 D08KQM 24816375 Ki = 149 nM T63179 D09OKK 9951771 IC50 < 20 nM T63179 D0F1SS 44605900 IC50 > 3000000 nM T63179 D0G5OV 11543746 IC50 = 3700 nM T63179 D0M0RS 11560224 Ki > 1000 nM T63179 D0V4RZ 25113722 IC50 > 10000 nM T63179 D0XS0R 44433505 Ki = 124 nM T28413 D0E3TC 44259 IC50 = 31.9 nM T28413 D0O6WV 24794418 IC50 > 500 nM T28413 D0T3ME 156422 IC50 = 1200 nM T28413 C5GE7T 9917045 IC50 = 3200 nM T28413 CUJR40 10062694 EC50 = 2 nM T28413 CSGD16 10246246 IC50 = 7000 nM T28413 C45EWD 11723489 IC50 = 8000 nM T28413 C6JV7W 23400934 IC50 > 7000 nM T28413 CD5S7O 23401001 IC50 = 9000 nM T28413 C7YG1N 24759534 IC50 = 180 nM T28413 C8B6TY 42628503 EC50 < 500 nM T28413 C3VRO9 44557921 IC50 > 10000 nM T28413 C8NA4L 53384644 IC50 > 30000 nM T28413 CJ47MX 56963907 IC50 > 10000 nM T28413 C9L6FD 56963908 IC50 > 10000 nM T28413 CE50IB 56963909 IC50 > 10000 nM T28413 CXJ63M 59603829 IC50 = 52 nM T28413 CQEU96 59603842 IC50 = 22 nM T28413 CV63UL 67240318 IC50 > 10000 nM T28413 C5DGR9 69036886 IC50 = 2094 nM T28413 C82FIP 70686752 IC50 = 3700 nM T28413 C0QX3Y 70688829 IC50 = 1600 nM T28413 CSOT12 70693058 IC50 > 10000 nM T28413 CS6NW3 70693059 IC50 > 10000 nM T28413 C1HW4B 89735655 IC50 > 100000 nM T28413 C9WGB8 127035904 IC50 = 3500 nM T28413 C7TG3J 137641313 IC50 > 19952.62 nM T28413 C2MD1Q 155513187 IC50 > 10000 nM T28413 D02BXJ 46864270 IC50 = 1.2 nM T28413 D05FXD 44478401 IC50 = 40 nM T28413 D0Q0YV 24944925 IC50 > 19952.62 nM T28413 D0R2WK 16038120 EC50 > 1000 nM T28413 D0X8BU 71718651 IC50 = 2500 nM T90751 C38SOR 71602434 IC50 = 63.1 nM T90751 C3ZR8K 71603028 IC50 = 501.19 nM T90751 CP97OC 71603093 IC50 = 50.12 nM T90751 CAHY94 71603095 IC50 = 158.49 nM T90751 C3IHF5 71603097 IC50 = 31.62 nM T90751 C9D1QC 71603211 IC50 = 398.11 nM T90751 CJTR16 71766152 IC50 > 50000 nM T90751 C8HN7U 122189249 IC50 > 40000 nM T90751 CNV03S 122189255 IC50 = 14900 nM T90751 C4MQU9 145980134 IC50 > 50000 nM T98293 D0R0MW 5329102 Ki = 500 nM T98293 D02RJY 11442891 IC50 > 10000 nM T98293 D03HUX 49792852 IC50 > 10000 nM T98293 D05ADP 160355 IC50 = 6900 nM T98293 D06KTJ 53252276 IC50 = 76 nM T98293 D08MHM 25227462 Ki = 15 nM T98293 D0E3TC 44259 IC50 = 1.9 nM T98293 D0MS3Z 16725726 IC50 = 10 nM T98293 D0O0LS 25141092 IC50 > 10000 nM T98293 D0P1CV 46191454 IC50 > 10000 nM T98293 D0Q9UX 16718576 IC50 > 10000 nM T98293 D0T3ME 156422 IC50 > 30000 nM T98293 C1ZG2U 449087 IC50 > 10000 nM T98293 CRB15U 521106 IC50 > 10000 nM T98293 C3J7LB 2951910 IC50 = 14.9 nM T98293 C24CDJ 10111591 IC50 = 790 nM T98293 C7HBP6 10429593 IC50 > 10000 nM T98293 CEML49 10538870 IC50 > 100000 nM T98293 C9O2PG 10588346 IC50 > 100000 nM T98293 C7KF2E 10705154 IC50 > 100000 nM T98293 C2C8GH 10732141 IC50 > 100000 nM T98293 CBOP58 11293798 Ki > 10000 nM T98293 CRTG16 11359538 IC50 > 20000 nM T98293 C26BZX 11362471 Ki > 10000 nM T98293 CWXB93 11397177 Ki > 10000 nM T98293 CTG83F 11539329 Ki > 5500 nM T98293 CMIL86 11590363 Ki > 5500 nM T98293 C9T6SC 11640926 Ki > 5500 nM T98293 C4GTZ8 11645322 IC50 > 20000 nM T98293 C9JT4S 11847343 IC50 = 455 nM T98293 C0ZWP3 15953852 Ki = 2 nM T98293 CFPW41 16007116 Ki > 5400 nM T98293 CZHJ34 16058637 IC50 = 5500 nM T98293 C5VPH9 16129448 IC50 = 46 nM T98293 CDO7W8 16202256 EC50 = 9 nM T98293 C1FC4H 21939235 Ki = 49 nM T98293 CF5SP7 24765704 EC50 = 36 nM T98293 C3W5AN 24765897 EC50 = 28 nM T98293 CI70UD 24765900 Ki = 30 nM T98293 C0VZQ5 24765998 EC50 = 4 nM T98293 C4EG8R 24993189 IC50 > 10000 nM T98293 CB21XV 25164469 Ki > 3750 nM T98293 CNF0A8 25164674 Ki > 3750 nM T98293 CUX83H 25164675 Ki > 3750 nM T98293 C1H7BF 25164677 Ki > 3750 nM T98293 CN50EI 25164678 Ki > 3750 nM T98293 C3XI7P 25164880 Ki > 3750 nM T98293 CX80QK 25164883 Ki > 3750 nM T98293 C6SD2A 25165081 Ki > 3750 nM T98293 C67TVH 25165085 Ki > 3750 nM T98293 C8J4KL 25165278 Ki = 3588 nM T98293 CRJ6M7 25165279 Ki > 3750 nM T98293 C7RBX0 25165280 Ki > 3750 nM T98293 CPEY29 25165481 Ki > 3750 nM T98293 C70DRX 25165482 Ki > 3750 nM T98293 CE8D1W 25165860 Ki = 69911 nM T98293 C6VZU2 25165861 Ki > 5450 nM T98293 C9VA1N 25166056 Ki = 13090 nM T98293 CX8HY9 25166657 Ki = 67636 nM T98293 CF4G1L 25167074 Ki > 3750 nM T98293 C35ZXL 25167075 Ki > 3750 nM T98293 C1CRJ7 25167076 Ki > 3750 nM T98293 C1IFX5 25167077 Ki > 3750 nM T98293 C2D3FP 25167078 Ki > 3750 nM T98293 CP2W8I 25167079 Ki > 3750 nM T98293 CJO5A4 25167275 Ki > 3750 nM T98293 C5KX0G 25167277 Ki > 3750 nM T98293 CQ5FJ8 25167278 Ki > 3750 nM T98293 C37YSX 25167280 Ki > 3750 nM T98293 CNG96H 25210579 IC50 > 10000 nM T98293 CB0O2A 44186880 Ki > 3750 nM T98293 C9K7OP 44186882 Ki > 3750 nM T98293 CX0ZU8 44186885 Ki > 3750 nM T98293 CNGV37 44189584 Ki > 3750 nM T98293 CGI5L7 44405938 IC50 > 20000 nM T98293 C0G3WF 44405939 IC50 > 20000 nM T98293 CR3Q7Z 44405940 IC50 > 20000 nM T98293 C79WRL 44405941 IC50 > 20000 nM T98293 C9ZNA0 44405945 IC50 > 100000 nM T98293 C9LD2T 44405946 IC50 > 100000 nM T98293 C0RO6U 44405949 IC50 = 13000 nM T98293 C2CTN7 44405982 IC50 > 100000 nM T98293 C0CR1O 44405983 IC50 = 37000 nM T98293 CW86VI 44405987 IC50 > 100000 nM T98293 C5V4TQ 44405999 IC50 > 100000 nM T98293 C0XZ8K 44406013 IC50 > 20000 nM T98293 CS3K1P 44406014 IC50 > 20000 nM T98293 CC93JP 44406018 IC50 > 20000 nM T98293 C7P0IH 44406019 IC50 > 20000 nM T98293 C4X2ME 44406047 IC50 > 100000 nM T98293 C36YDV 44406048 IC50 > 100000 nM T98293 CXZ5C3 44406055 IC50 > 100000 nM T98293 CCRZ12 44406074 IC50 > 20000 nM T98293 CZ1R8M 44450033 IC50 > 100000 nM T98293 CIY3T5 44450035 IC50 > 100000 nM T98293 C5Y4PN 44450059 IC50 > 100000 nM T98293 C28LMV 44450060 IC50 > 100000 nM T98293 C3VRO9 44557921 IC50 = 9332.54 nM T98293 CU3RF1 45139989 IC50 > 10000 nM T98293 CQGZ06 45139991 IC50 > 10000 nM T98293 CY3HW5 46224684 IC50 = 2300 nM T98293 C7ON5A 46233287 IC50 > 10000 nM T98293 CLS29B 46872626 IC50 > 10000 nM T98293 C2O8RZ 46886323 IC50 > 1000 nM T98293 C52OJN 47052811 IC50 = 8700 nM T98293 CF91RS 49843531 IC50 > 10000 nM T98293 C2Y6QS 50938552 IC50 > 10000 nM T98293 C9NYP4 51036677 IC50 > 10000 nM T98293 C4WRY3 51037112 IC50 > 10000 nM T98293 CRI28Z 51037948 IC50 > 10000 nM T98293 CDU4Q5 51346827 Ki > 3750 nM T98293 CZS8K4 53319042 Ki > 3750 nM T98293 CUD21V 53320263 Ki > 3750 nM T98293 CESA85 53323614 Ki > 3750 nM T98293 C8NA4L 53384644 IC50 > 30000 nM T98293 CE1ZK6 54759168 IC50 > 10000 nM T98293 CBOD63 56835089 IC50 > 30000 nM T98293 CD6Y9Z 57395116 IC50 > 30000 nM T98293 C8W6IG 57395117 IC50 > 30000 nM T98293 CG7S0D 57396882 IC50 > 30000 nM T98293 C0C7ET 57523203 EC50 < 1 nM T98293 CD51JZ 57523643 Ki = 64 nM T98293 C69JRB 57523678 Ki = 512 nM T98293 C7OSL3 57523679 EC50 = 21 nM T98293 C2GV3D 57523680 EC50 = 11 nM T98293 CC8N1R 57523705 EC50 = 15 nM T98293 CJ2H3Y 57523706 EC50 = 16 nM T98293 CKG45N 57523707 EC50 = 18 nM T98293 CZXT03 57523708 EC50 = 1 nM T98293 CCX16J 57523709 EC50 = 7 nM T98293 CE12XV 60163664 Ki = 670 nM T98293 C6DUK0 60163745 Ki = 68 nM T98293 C8BV6Z 60163908 Ki = 120 nM T98293 CDYE40 60164283 Ki = 1300 nM T98293 CCUH92 60164742 Ki = 600 nM T98293 C4GK3V 60164846 Ki = 32 nM T98293 C37NKO 67129970 IC50 = 6440 nM T98293 CK80LJ 67130050 IC50 = 6790 nM T98293 CV63UL 67240318 IC50 > 10000 nM T98293 C12DPO 68060125 IC50 = 779 nM T98293 C36BVQ 68181618 Ki > 2900 nM T98293 CUQ4F0 68181642 Ki > 2900 nM T98293 CAN7U2 68181681 Ki > 2900 nM T98293 CK7XJ5 68181838 Ki = 140 nM T98293 CFQ9N0 68181876 Ki > 2900 nM T98293 C4VK1Q 68181882 Ki > 2900 nM T98293 CQC0R5 68181954 Ki = 3.3 nM T98293 C7GRV2 68755406 IC50 > 10000 nM T98293 C82YNL 70934541 IC50 > 10000 nM T98293 CQA4U7 71528975 Ki = 272 nM T98293 CCN01X 71547862 IC50 > 10000 nM T98293 C1NPL0 71552941 IC50 > 30000 nM T98293 CA4PS8 71552942 IC50 > 30000 nM T98293 C3UA9C 71553011 IC50 = 30000 nM T98293 CEZ15Y 71553012 IC50 = 30000 nM T98293 CVIA91 71553085 IC50 = 30000 nM T98293 C1TR3O 71553152 IC50 = 30000 nM T98293 CRX81Q 71575642 IC50 > 10000 nM T98293 CH97AJ 71611283 Ki = 505 nM T98293 C0OPM4 72725813 Ki = 60 nM T98293 CWK65Y 76329224 Ki = 190 nM T98293 C9M6JR 76332879 Ki = 500 nM T98293 CUF60Q 86274945 IC50 = 5.3 nM T98293 C49LZW 89766055 Ki = 1300 nM T98293 CHI39S 90292823 IC50 = 673 nM T98293 CY0UC4 90645194 IC50 > 10000 nM T98293 C6Y4PV 91809512 Ki = 12 nM T98293 C8Y2GZ 91809513 Ki = 4 nM T98293 CY7BI2 118706214 IC50 > 10000 nM T98293 CIM4B7 118720596 IC50 = 35.5 nM T98293 C01QJE 122178550 Ki = 45 nM T98293 C87ERY 122178551 Ki = 283 nM T98293 C30LEZ 122178552 Ki = 612 nM T98293 C4NSI0 122178553 Ki = 1820 nM T98293 C41KSU 122178554 Ki = 80 nM T98293 C3BHS9 122178555 Ki = 100 nM T98293 CDUA42 122182198 Ki = 629 nM T98293 C30URY 122182199 Ki = 617 nM T98293 CNZG96 122182482 Ki > 2900 nM T98293 C9ENM4 122182483 Ki > 2900 nM T98293 CV3X7Z 122182484 Ki = 950 nM T98293 CV7E8D 122182485 Ki = 1270 nM T98293 CFP8L3 122182486 Ki = 344 nM T98293 C41VZY 122182487 Ki = 621 nM T98293 C9Z5AY 122182488 Ki = 2490 nM T98293 CSN1P8 122182489 Ki = 817 nM T98293 C74VXS 122182490 Ki = 1020 nM T98293 CL3PR1 122182491 Ki > 2900 nM T98293 CQ8XC0 122183105 IC50 = 1200 nM T98293 C3C5DB 122183106 IC50 = 550 nM T98293 C4D6UX 122183107 IC50 = 170 nM T98293 C7GO9K 122183108 IC50 > 10000 nM T98293 C4X7SD 122192466 IC50 > 10000 nM T98293 CK6YP3 132274772 Ki = 51 nM T98293 CJ9D8A 132274773 Ki = 710 nM T98293 C9GS1O 132502974 IC50 = 27 nM T98293 C52FCI 134817245 Ki = 28 nM T98293 CMB4C1 135198759 Ki = 354 nM T98293 CS90MD 135198762 Ki = 3890 nM T98293 C8NC5Z 135198764 Ki = 672 nM T98293 C35GVJ 135198767 Ki = 3817 nM T98293 C5AK2R 135198771 Ki = 114 nM T98293 CD85HP 135198778 Ki = 45 nM T98293 C5BY1N 135198783 Ki = 768 nM T98293 C19BPG 135198785 Ki = 2172 nM T98293 CFI13G 135198787 Ki = 16 nM T98293 CQUW03 135198795 Ki = 306 nM T98293 CGJ4P7 135198796 Ki = 151 nM T98293 C3AP4K 135198799 Ki = 6 nM T98293 CFT06G 135198805 Ki = 2408 nM T98293 C3VX2F 135198838 Ki = 119 nM T98293 CNJT83 135198992 Ki = 674 nM T98293 CEML07 135199057 Ki = 17 nM T98293 CU60YC 135431661 IC50 = 14370 nM T98293 CHA4N2 136013680 IC50 > 10 nM T98293 CM5T4K 136176135 Ki = 6 nM T98293 C6H4CY 136176136 Ki = 2.8 nM T98293 C1YUD0 136219394 IC50 > 10 nM T98293 CIU8W3 136254389 IC50 > 10 nM T98293 CV6WC3 137348710 Ki = 9 nM T98293 CBYQ40 137631877 IC50 = 1056 nM T98293 CT15UJ 137632050 IC50 = 483 nM T98293 C8ES9F 137632070 IC50 = 1423 nM T98293 CO9J0E 137632679 IC50 = 379 nM T98293 CGQZ93 137632703 Ki = 36 nM T98293 CHO1X9 137633641 IC50 = 4470 nM T98293 CS67LW 137633708 IC50 = 3376 nM T98293 CN17FY 137633916 IC50 > 10000 nM T98293 CI1E8V 137634241 IC50 > 10000 nM T98293 C8S7YK 137634619 Ki = 26 nM T98293 CWZ91Y 137634945 IC50 = 1163 nM T98293 C5S7PK 137635580 Ki = 16 nM T98293 C5HP6C 137635864 Ki = 77 nM T98293 COQ9B3 137636317 IC50 = 1736 nM T98293 CX7W5Q 137636419 IC50 = 1709 nM T98293 CR2O8C 137638015 IC50 = 1987 nM T98293 CB5V3J 137638022 IC50 = 1255 nM T98293 CW0IV9 137638647 Ki = 1440 nM T98293 CJ3PT6 137639406 IC50 = 5005 nM T98293 CM0B1F 137640432 Ki = 576 nM T98293 CN7O5H 137640572 IC50 = 54 nM T98293 C64SKI 137640706 IC50 = 304 nM T98293 C3X7SM 137641415 Ki = 11 nM T98293 C5RT8G 137641563 IC50 = 33 nM T98293 C5LC9F 137642132 IC50 = 93 nM T98293 C39QYI 137642461 IC50 = 1506 nM T98293 C4Z8QM 137643488 IC50 = 1454 nM T98293 CAJV07 137643540 IC50 = 3956 nM T98293 CMZ8T5 137643638 Ki = 782 nM T98293 CZNP51 137644346 IC50 = 1290 nM T98293 CXV64J 137644569 IC50 = 1201 nM T98293 CAO28T 137644956 Ki = 99 nM T98293 C7QF2S 137645076 IC50 = 937 nM T98293 CF2IP5 137645363 IC50 = 634 nM T98293 CN9HO2 137645749 IC50 = 788 nM T98293 C4PDY1 137646859 IC50 = 3071 nM T98293 C1LSX3 137647136 IC50 = 802 nM T98293 CXJQ26 137648567 Ki = 7 nM T98293 C1B4LS 137649300 Ki = 16 nM T98293 CP4Z0J 137651385 Ki = 1630 nM T98293 CCB7J9 137651438 Ki = 325 nM T98293 CN1ET2 137651558 IC50 = 177 nM T98293 C4QOD8 137651940 IC50 = 16 nM T98293 C8H6DO 137652195 IC50 = 2040 nM T98293 C65OIK 137652229 IC50 = 391 nM T98293 C8SV7X 137653128 Ki = 218 nM T98293 CBA6H2 137653619 IC50 = 920 nM T98293 CPW29A 137654589 IC50 = 281 nM T98293 C7QF9U 137655545 IC50 = 3145 nM T98293 COH17C 137655886 IC50 = 718 nM T98293 CN3TV9 137655924 IC50 = 2334 nM T98293 C3M4JV 137656092 Ki = 256 nM T98293 C9HD5U 137656968 IC50 = 406 nM T98293 CH3EI4 137657621 IC50 = 633 nM T98293 CXU27T 137657885 IC50 = 22 nM T98293 CT50JU 137658259 IC50 = 360 nM T98293 CS89BI 137658282 IC50 = 1544 nM T98293 CCL9G1 137659229 IC50 = 3516 nM T98293 CXK23M 137659630 Ki = 17 nM T98293 CGL65U 137659799 IC50 = 2355 nM T98293 CNF2G3 137659831 IC50 = 199 nM T98293 C1FI8B 137659938 Ki = 884 nM T98293 CTP7A3 137660199 IC50 = 1757 nM T98293 CT4FA3 137662174 Ki = 652 nM T98293 CI9YB7 138753112 IC50 = 25 nM T98293 C6VB3O 145925651 IC50 >= 5000 nM T98293 C7XPB3 145949197 IC50 = 114 nM T98293 C1M8VJ 145949527 IC50 = 323 nM T98293 C2DZ9Q 145949981 IC50 = 530 nM T98293 CU1M5G 145950938 IC50 = 67 nM T98293 CW50LC 145951514 IC50 = 63 nM T98293 C8UG3Q 145952059 IC50 > 10000 nM T98293 CX71CV 145952439 IC50 > 10000 nM T98293 CF4NM5 145952455 IC50 = 61 nM T98293 CR5C3F 145952528 IC50 = 89 nM T98293 CY04AZ 145952979 IC50 = 115 nM T98293 CW04QR 145953124 IC50 = 3285 nM T98293 C7ZA2L 145953846 IC50 = 689 nM T98293 CLI14F 145954605 IC50 > 10000 nM T98293 C6VX9D 145954723 IC50 = 270 nM T98293 CO3V9N 145957397 IC50 = 1112 nM T98293 CN9L8K 145957820 IC50 = 32 nM T98293 C6OZ8V 145958048 IC50 = 4212 nM T98293 CBZ84P 145958367 IC50 > 10000 nM T98293 CZN93D 145959664 IC50 = 706 nM T98293 C9O4EX 145959847 IC50 > 10000 nM T98293 CH5XC4 145959996 IC50 = 139 nM T98293 CK75RE 145960054 IC50 = 621 nM T98293 CY4HO8 145971464 IC50 = 410 nM T98293 C2WOG0 145973860 IC50 = 162 nM T98293 C2MD1Q 155513187 IC50 > 10000 nM T98293 D00ERW 44444843 Ki > 5454 nM T98293 D00HVA 11624601 Ki > 5500 nM T98293 D03DZO 11715767 IC50 > 10000 nM T98293 D07OAT 456214 IC50 = 130 nM T98293 D08HFG 24809764 IC50 > 10000 nM T98293 D09HVH 135566652 IC50 > 10 nM T98293 D0F0AU 44405988 IC50 > 20000 nM T98293 D0O6OH 71553154 IC50 = 5720 nM T98293 D0Q3NG 11715520 Ki > 5500 nM T98293 D0S7IE 11658882 Ki > 5500 nM T98293 D0T8NU 16757525 IC50 > 4000 nM T58470 D06WHY 16747683 IC50 = 45 nM T58470 CU94SN 447671 IC50 = 680 nM T58470 CKU98Q 447672 IC50 = 5600 nM T58470 C8UAE2 10124259 IC50 = 50 nM T58470 C3GC8T 11563920 IC50 = 530 nM T58470 CA7U1P 52940779 IC50 = 12000 nM T58470 CO4QZ1 52946827 IC50 = 21000 nM T58470 CZG8K0 52949286 IC50 = 590 nM T97413 D01XNB 4594 EC50 = 14000 nM T97413 CS24QK 155794 EC50 = 3900 nM T97413 CKM51L 1214469 EC50 = 440 nM T97413 C9DQV6 3288900 EC50 = 10000 nM T97413 C3WS7Q 4157547 EC50 = 220 nM T97413 C4M6VX 4254919 EC50 = 4525 nM T97413 CI8S7A 4581089 EC50 = 380 nM T97413 C7YA5T 4899895 EC50 = 10000 nM T97413 C36EBJ 4900723 EC50 = 10000 nM T97413 C60UTZ 6324606 EC50 = 4500 nM T97413 CU16RT 11891917 EC50 = 940 nM T97413 CCNL10 13909784 EC50 > 32000 nM T97413 CIVD51 25025858 EC50 = 106 nM T97413 CKQ07S 25025861 IC50 = 19 nM T97413 C9UA8V 25025862 IC50 = 33 nM T97413 CIC9V8 25025863 EC50 = 30 nM T97413 C9K1JE 25026044 IC50 = 11 nM T97413 C13KEJ 25026056 EC50 = 102 nM T97413 CACJ32 25026058 IC50 = 18 nM T97413 CNW89T 25026445 EC50 = 67 nM T97413 CL75TW 25026446 EC50 = 16 nM T97413 CJS39H 25055504 IC50 = 82 nM T97413 CENH94 25110720 EC50 = 510 nM T97413 CA1KD6 25128865 IC50 = 1.6 nM T97413 CLXT92 25128867 EC50 = 82 nM T97413 CJE98Q 25129212 IC50 = 0.5 nM T97413 C78RUM 25134006 IC50 = 8.3 nM T97413 CQHC91 25134007 IC50 = 1.7 nM T97413 COFC90 25249151 EC50 = 10000 nM T97413 CNK9I6 44300265 EC50 = 0.19 nM T97413 CEG32A 44300275 EC50 = 30 nM T97413 CND1W8 44300286 EC50 = 151 nM T97413 CIM97P 44300355 EC50 = 1.4 nM T97413 CZE85M 44300356 EC50 = 3.1 nM T97413 C0MX2R 44300379 EC50 = 2.2 nM T97413 CRJ16V 44300383 EC50 = 7900 nM T97413 C5HMV8 44300407 EC50 = 6 nM T97413 CUN1C2 44300408 EC50 = 15 nM T97413 CMT21V 44300413 EC50 = 9.3 nM T97413 C26GDB 44300427 EC50 = 17 nM T97413 CR7S9A 44300429 EC50 = 21 nM T97413 CW5QR3 44300436 EC50 = 2.9 nM T97413 CXZ6W5 44300451 EC50 = 1.5 nM T97413 CL5T7N 44300456 EC50 = 240 nM T97413 CIUO48 44300482 EC50 = 2700 nM T97413 C3CE5F 44300503 EC50 = 70 nM T97413 CY6DH5 44300505 EC50 = 21 nM T97413 C8FU5P 44300796 EC50 = 24 nM T97413 CS01QY 44387452 EC50 = 19 nM T97413 CRS04C 44388192 IC50 = 1.1 nM T97413 CQI54O 44589789 EC50 > 32000 nM T97413 CH54CO 44589824 EC50 = 1600 nM T97413 C89LHN 44589825 EC50 > 32000 nM T97413 C9AC4P 44589826 EC50 > 32000 nM T97413 CCG7E4 44589827 EC50 > 32000 nM T97413 C9A7EH 44589871 EC50 > 32000 nM T97413 CG62MO 44589872 EC50 = 210 nM T97413 C23ODF 44589873 EC50 > 32000 nM T97413 CN50MX 44589874 EC50 = 350 nM T97413 CAPD56 44589875 EC50 > 32000 nM T97413 C6A9FB 44589925 EC50 > 32000 nM T97413 C3XF1Z 44589926 EC50 > 32000 nM T97413 CO7V1C 44589927 EC50 > 32000 nM T97413 CD29AO 44589928 EC50 = 570 nM T97413 CF8S6V 44589929 EC50 = 240 nM T97413 C4DXG0 44589930 EC50 > 32000 nM T97413 CIVJ75 44589982 EC50 > 32000 nM T97413 C7SW1I 44589983 Ki = 0.36 nM T97413 CJA6H8 46861857 EC50 = 41 nM T97413 CUC57I 46881416 EC50 = 205 nM T97413 CGM8U7 46881417 EC50 = 1323 nM T97413 C4NLI8 46881418 EC50 = 1724 nM T97413 CFP9M3 46881419 EC50 = 5479 nM T97413 CF10NE 46881470 EC50 = 812 nM T97413 CFYG76 46881471 EC50 = 127 nM T97413 C5K0XD 46881472 EC50 = 4307 nM T97413 C2A5NH 46881473 EC50 = 159 nM T97413 CKSV37 46881507 EC50 = 2663 nM T97413 CH2C3I 46881508 EC50 = 825 nM T97413 C5H9VN 46881509 EC50 = 2288 nM T97413 CA7F0L 46881510 EC50 = 177 nM T97413 C7RF0S 46881558 EC50 = 1601 nM T97413 COX74V 46881559 EC50 = 87 nM T97413 C1GCR2 46881560 EC50 = 1004 nM T97413 C7QT0J 46881561 EC50 = 588 nM T97413 CA26ZQ 46881601 EC50 = 41 nM T97413 C07DSX 46881602 EC50 = 88 nM T97413 C1X5LG 46881603 EC50 = 642 nM T97413 CZED45 46881604 EC50 = 375 nM T97413 CSA4G7 46881605 EC50 = 338 nM T97413 C0UC1I 46881642 EC50 = 119 nM T97413 C4CH6M 46881643 EC50 = 39 nM T97413 C3DZ2A 46881644 EC50 = 4334 nM T97413 C20EUS 46881683 EC50 = 76 nM T97413 C62ZHB 46881920 EC50 = 2722 nM T97413 C8BUD7 46881921 EC50 = 2760 nM T97413 CIY5R4 46881961 EC50 = 2707 nM T97413 C46YQV 46881962 EC50 = 4124 nM T97413 C9LQ6W 46881963 EC50 = 5360 nM T97413 CLT64X 46881964 EC50 = 5887 nM T97413 CCS3V2 46882010 EC50 = 292 nM T97413 C2G4YW 46882011 EC50 = 1897 nM T97413 COV81C 46882012 EC50 = 2656 nM T97413 C1AL2I 46882013 EC50 = 1183 nM T97413 C2BWN6 46882057 EC50 = 4618 nM T97413 CFAU65 46882058 EC50 > 10000 nM T97413 C40JVD 46882059 EC50 = 5598 nM T97413 C06SQX 46882060 EC50 = 4376 nM T97413 CDN0M6 46882061 EC50 = 4949 nM T97413 CX9KN4 46884576 EC50 = 98 nM T97413 C09YKP 46884577 EC50 = 98 nM T97413 C7Z8PM 46884578 EC50 = 95 nM T97413 CDBV62 46884627 EC50 = 100 nM T97413 C2JK0N 46884628 IC50 = 7.3 nM T97413 CLY46C 46884629 EC50 = 95 nM T97413 CF06QJ 46884630 IC50 = 11 nM T97413 C9DMF5 46884659 EC50 = 104 nM T97413 C1B8HE 46884660 EC50 = 44 nM T97413 C5R6CX 46884661 IC50 = 51 nM T97413 CZTW82 46884662 EC50 = 89 nM T97413 CXNW15 46884663 EC50 = 93 nM T97413 C8W6FA 46884687 EC50 = 89 nM T97413 CA2GZ0 46884688 EC50 = 108 nM T97413 CDE9R6 46885311 EC50 = 63 nM T97413 C17TDW 46885312 EC50 = 95 nM T97413 CY8S7V 46885313 EC50 = 15 nM T97413 C4P5TG 46887765 EC50 = 10000 nM T97413 CUV81Y 46887766 EC50 = 10000 nM T97413 CY19ZW 46887767 EC50 = 10000 nM T97413 C28YFQ 46887768 EC50 = 10000 nM T97413 C0BRH4 46887824 EC50 = 10000 nM T97413 CBL16I 46887825 EC50 = 10000 nM T97413 CEI50R 46887826 EC50 = 10000 nM T97413 C8N9DJ 46887875 EC50 = 10000 nM T97413 CBQH46 46887876 EC50 > 10000 nM T97413 CI9G1L 46887877 EC50 = 6779 nM T97413 C7Z2FK 46887912 EC50 = 5567 nM T97413 CL82BA 46887914 EC50 = 10000 nM T97413 CWH39F 46887915 EC50 = 10000 nM T97413 C73ZFT 46887916 EC50 = 10000 nM T97413 CV9I3H 46887946 EC50 = 10000 nM T97413 C0OKC5 46887947 EC50 = 10000 nM T97413 COF5Z1 46887948 EC50 = 10000 nM T97413 CO25LZ 46887949 EC50 = 10000 nM T97413 C71EUT 46887950 EC50 = 10000 nM T97413 CMN5W7 46887979 EC50 > 10000 nM T97413 CU38HW 46887980 EC50 = 3164 nM T97413 C63KXC 46887981 EC50 = 3474 nM T97413 C96XQN 46887982 EC50 = 4763 nM T97413 CPNK87 46888017 EC50 = 1542 nM T97413 C6B9LH 46888018 EC50 = 1234 nM T97413 CUH5F2 46888019 EC50 = 704 nM T97413 CN8D6R 46888020 EC50 = 543 nM T97413 C8JPX1 46888066 EC50 = 10000 nM T97413 C12JRM 46888067 EC50 = 4149 nM T97413 CLJY59 46888068 EC50 = 10000 nM T97413 CV78GQ 46888069 EC50 = 10000 nM T97413 C4FN7U 46889145 EC50 = 56 nM T97413 C3Z2OS 46889146 EC50 = 133 nM T97413 CD17TV 46889148 EC50 = 54 nM T97413 C2LOX3 46889175 EC50 = 172 nM T97413 C1FHB0 46889176 EC50 = 78 nM T97413 C5H3ID 46889177 EC50 = 129 nM T97413 C9W1TE 46889209 IC50 = 83 nM T97413 COC75X 46889210 EC50 = 29 nM T97413 C7RFY6 46889232 IC50 = 20 nM T97413 CB7QS5 46889233 IC50 = 5.3 nM T97413 CU02WV 46889234 IC50 = 6.2 nM T97413 CW4JV1 46889235 IC50 = 26 nM T97413 CLM87T 53242205 EC50 = 55 nM T97413 CF46OQ 54580461 EC50 = 51 nM T97413 CO2D3K 54580462 EC50 = 350 nM T97413 CW09DM 54580463 EC50 = 450 nM T97413 CZ0X6O 54580464 EC50 > 10000 nM T97413 C7HLQ4 54580465 EC50 = 8100 nM T97413 CH7D2O 54581470 EC50 = 160 nM T97413 CPY2S1 54581471 EC50 = 220 nM T97413 C37JZI 54581472 EC50 = 6400 nM T97413 CBNF48 54581473 IC50 = 9700 nM T97413 CTA0N4 54581474 EC50 = 4000 nM T97413 CON1G8 54581475 EC50 = 10000 nM T97413 CRY30T 54582477 EC50 = 2100 nM T97413 CPB58V 54582478 IC50 = 310 nM T97413 CL0S1D 54583450 IC50 = 3800 nM T97413 CSB32Y 54583451 EC50 = 8300 nM T97413 CNM94E 54583452 EC50 = 2600 nM T97413 C2DJ8T 54583453 EC50 = 4000 nM T97413 C5SGL3 54583454 EC50 = 1200 nM T97413 CQ3W9F 54584418 EC50 = 720 nM T97413 CWXZ37 54584419 EC50 > 10000 nM T97413 C6I7DX 54584420 EC50 = 8300 nM T97413 CKI26O 54584421 EC50 = 8200 nM T97413 CZ6T8E 54585379 EC50 = 1200 nM T97413 C0RMX2 54585380 EC50 = 640 nM T97413 C5YQ4V 54586335 EC50 = 1700 nM T97413 CPY6T7 54586336 EC50 = 7500 nM T97413 CEJ51B 54586337 EC50 = 1600 nM T97413 CY7LG4 54587369 IC50 = 400 nM T97413 CZU39D 59618620 EC50 = 110 nM T97413 C9EWC4 59618623 IC50 = 6.8 nM T97413 CPUV97 59618635 IC50 = 10 nM T97413 CF8IM7 59618646 IC50 = 40 nM T97413 CX8H6V 59618658 IC50 = 14 nM T97413 C28OWH 59618675 IC50 = 20 nM T97413 CVF85X 59618678 IC50 = 4.4 nM T97413 C0IO7P 59618681 EC50 = 108 nM T97413 C8B4JL 59618698 EC50 = 43 nM T97413 CXK59H 59618709 EC50 = 38 nM T97413 CF8AT2 59618710 EC50 = 277 nM T97413 CBO13Y 59618711 IC50 = 2.1 nM T97413 CYH7R9 59618730 EC50 = 60 nM T97413 CT8M5F 59618746 IC50 = 0.5 nM T97413 CAKY62 59618747 EC50 = 42 nM T97413 C8UJ7N 59618753 IC50 = 0.7 nM T97413 CZ3J1K 59618778 EC50 = 543 nM T97413 CK9Z8R 59618785 IC50 = 10 nM T97413 CEU67L 59618790 IC50 = 0.9 nM T97413 CBFA01 59618811 EC50 = 110 nM T97413 CW0UD7 59618821 IC50 = 1.4 nM T97413 CWR3U0 62707207 IC50 = 18 nM T97413 CV4BD2 62707362 IC50 = 0.76 nM T97413 CYU24M 62707363 IC50 = 1.4 nM T97413 CXD5M1 62707364 IC50 = 1.1 nM T97413 C8SKU9 62707365 IC50 = 1.2 nM T97413 C2E0YG 62707528 IC50 = 1.9 nM T97413 C0L5QH 66901749 EC50 = 50 nM T97413 CQO03N 66901760 EC50 = 63 nM T97413 C1V5BY 71451943 EC50 > 10000 nM T97413 C64UGX 71451990 IC50 = 5 nM T97413 CN2PK3 71451991 EC50 = 88 nM T97413 C75QOT 71460937 EC50 = 69 nM T97413 CXG62J 71460964 EC50 = 199 nM T97413 C94VXI 71462686 IC50 = 430 nM T97413 CJC7E2 73345589 IC50 > 100 nM T97413 C5X1KD 73351696 IC50 > 100 nM T97413 CCN5K8 76310617 EC50 = 70 nM T97413 C5T0HJ 76310618 EC50 > 10000 nM T97413 C2YA1R 76310619 EC50 = 25 nM T97413 CMW68G 76314245 EC50 = 8.1 nM T97413 CT3B2I 76314246 EC50 = 368 nM T97413 CBC8E4 76314247 EC50 = 1.3 nM T97413 C6SWI3 76317820 EC50 = 2041 nM T97413 CRYK15 76317821 EC50 = 41 nM T97413 C2DIX3 76317822 EC50 = 48 nM T97413 C8RL4G 76317823 EC50 = 254 nM T97413 CY8L3Z 76321531 EC50 = 1562 nM T97413 C7W3MU 76321532 EC50 = 1.6 nM T97413 CP83JR 76325132 EC50 = 9.5 nM T97413 C4H8QK 76325133 EC50 = 12 nM T97413 C4B0TY 76325134 EC50 = 17 nM T97413 CWF9U5 76325135 EC50 = 8.5 nM T97413 C8Q5ZW 76328694 EC50 = 916 nM T97413 CLG24P 76328695 EC50 = 381 nM T97413 C0FR9H 76328696 EC50 = 11 nM T97413 C29XJO 76328697 EC50 = 13 nM T97413 C6H7JU 76328698 EC50 = 1.7 nM T97413 CMH01Z 76328699 EC50 = 6.9 nM T97413 C75OIT 76332370 EC50 = 131 nM T97413 CXY3G2 76332371 EC50 = 977 nM T97413 C63OMG 76332372 EC50 = 2046 nM T97413 CZ6J7Y 76332373 EC50 = 2071 nM T97413 CZ0XQ6 76336000 EC50 = 156 nM T97413 C2JN6K 76336001 EC50 = 59 nM T97413 CP7R4H 76336002 EC50 = 199 nM T97413 CXQ76V 76336003 EC50 = 4378 nM T97413 C2AT5Z 76336004 EC50 = 6.8 nM T97413 C73XHA 76336005 EC50 = 3.6 nM T97413 CS4ZG6 90663956 EC50 = 140 nM T97413 CRD81Y 90663957 EC50 = 79 nM T97413 CJV6C7 90663958 EC50 = 25 nM T97413 C9Q8SD 90663959 EC50 = 4 nM T97413 CRPV47 90663960 EC50 = 7.8 nM T97413 CIK0W5 90663961 EC50 = 6400 nM T97413 CRHU68 90663962 EC50 = 46 nM T97413 CN8EJ0 90663963 EC50 = 310 nM T97413 C9R6EX 90663964 EC50 = 710 nM T97413 CLZ7J2 90663965 EC50 = 1400 nM T97413 CFCD64 90663966 EC50 = 57 nM T97413 COBI56 90663967 EC50 = 32 nM T97413 CPV9L5 90663968 EC50 = 2.1 nM T97413 C9S6FN 90663969 EC50 = 230 nM T97413 CC5J7U 90663970 EC50 = 1200 nM T97413 CDNM68 118721521 EC50 > 10000 nM T97413 C4NH5Z 118721522 EC50 = 68 nM T97413 CF84QS 118721523 EC50 = 19 nM T97413 CVY85D 118721524 EC50 = 42 nM T97413 C9D6HQ 118721525 EC50 = 8.7 nM T97413 CPJZ65 118721526 EC50 > 10000 nM T97413 CKR9J4 118721527 EC50 = 40 nM T97413 CXJ3C5 118721528 EC50 = 4.2 nM T97413 CTM3L0 118721529 EC50 = 4 nM T97413 CV31RB 118721530 EC50 = 3.4 nM T97413 C4UQ8L 118721531 EC50 = 5.6 nM T97413 C40DIV 132538074 EC50 = 39 nM T97413 CBN97X 136086809 EC50 = 336 nM T97413 CQJ20H 136118727 EC50 = 77 nM T97413 CX6E8P 155511392 EC50 = 0.9 nM T97413 CGX15T 155515849 EC50 > 10000 nM T97413 C4J9CZ 155519281 EC50 = 2 nM T97413 CDC4R0 155519753 EC50 = 2230 nM T97413 C1OD0X 155520679 EC50 = 42 nM T97413 C86WTX 155521672 EC50 = 11 nM T97413 CL9F7G 155528415 EC50 = 1 nM T97413 CR34LQ 155530555 EC50 = 11 nM T97413 CL69NV 155538227 EC50 = 69 nM T97413 CMT4J7 155539847 EC50 = 21 nM T97413 C4KAU2 155541223 EC50 = 4085 nM T97413 C7YA6U 155543657 EC50 = 12 nM T97413 CJ2PT5 155543793 EC50 = 968 nM T97413 C94MFI 155552947 EC50 = 644 nM T97413 CB1D0U 155554592 EC50 = 13 nM T97413 C90ZVP 155557839 EC50 > 10000 nM T97413 CB3KQ9 155561529 EC50 = 3 nM T97413 CRAY42 155568183 EC50 = 897 nM T97413 C2Z9RC 155568881 EC50 = 3 nM T97413 D02TPY 25025860 EC50 = 47 nM T97413 D04JSE 46200989 EC50 = 1.4 nM T97413 D08RQW 49871766 Ki = 3.7 nM T97413 D0A0DS 25025654 EC50 = 133 nM T97413 D0A1FE 91827364 EC50 = 12 nM T97413 D0H4LP 72944991 EC50 = 1.7 nM T97413 D0MH6P 11434815 IC50 > 100 nM T97413 D0R8TG 11389266 IC50 = 37 nM T97413 D0T9VC 56840673 IC50 = 1.4 nM T97413 D0U4ZS 46845425 IC50 = 11 nM T09826 D02PMO 60700 IC50 = 21 nM T09826 D07VLY 31703 IC50 = 20000 nM T09826 D0B7EB 36462 IC50 > 1000000 nM T09826 D0H3WI 37542 IC50 = 65880 nM T09826 D0H4JM 8969 IC50 = 30000 nM T09826 D0J4JM 5770 IC50 = 160000 nM T09826 D0Z4XW 60699 IC50 = 1080 nM T09826 D07UHX 72402 IC50 = 110 nM T09826 D09YDM 24360 IC50 = 25 nM T09826 D0I1DW 9808998 EC50 = 51 nM T09826 D0ND9T 184196 IC50 > 30000 nM T09826 D0B3CT 9928668 EC50 > 3000 nM T09826 D0Q7FC 60956 IC50 = 416 nM T09826 CIX3P6 2538 IC50 = 1400 nM T09826 CKWN79 72403 IC50 = 30 nM T09826 CX4YM1 72486 IC50 = 4.2 ug.mL-1 T09826 CKH0W1 73170 IC50 > 250000 nM T09826 CUPX10 80427 IC50 > 100000 nM T09826 CPMU27 104986 IC50 = 140 nM T09826 C37VTK 123614 EC50 = 270 nM T09826 C02ABV 131182 IC50 = 440 nM T09826 C5O9RJ 165798 EC50 > 100000 nM T09826 CR1JW2 231860 IC50 > 100000 nM T09826 C7Y0CH 238747 IC50 > 200000 nM T09826 CD7VE0 366358 IC50 = 38 nM T09826 C5D8KX 368336 IC50 = 570 nM T09826 C5F2WA 419666 IC50 = 60000 nM T09826 CCK68G 441921 IC50 > 250000 nM T09826 C5DL0V 468669 IC50 = 48 nM T09826 CHA3Z1 468670 IC50 = 15 nM T09826 CYMH94 471008 IC50 = 106000 nM T09826 C0IJV9 486154 IC50 > 30000 nM T09826 C97MEG 494163 IC50 = 1600 nM T09826 CXD5F2 496192 IC50 > 200000 nM T09826 C82EPK 637517 IC50 > 1000000 nM T09826 CCIW48 694275 EC50 = 48950 nM T09826 CLJM48 697030 EC50 > 100000 nM T09826 CN7P9V 710216 EC50 > 100000 nM T09826 C10UJN 717415 EC50 > 100000 nM T09826 CY3FQ6 722747 EC50 > 100000 nM T09826 CH05JG 743742 EC50 = 93200 nM T09826 C4AE2I 760516 EC50 > 100000 nM T09826 CP6TJ4 840074 EC50 > 100000 nM T09826 CJW6V8 1277565 EC50 > 100000 nM T09826 COY89G 3738100 IC50 = 6100 nM T09826 CVQY83 3755712 IC50 = 47530 nM T09826 CX32RQ 5810410 EC50 > 100000 nM T09826 C5EAM3 6335134 IC50 > 30000 nM T09826 C0XKU9 6382696 EC50 > 100000 nM T09826 CT2C8S 6620659 IC50 > 100000 nM T09826 CR3ID2 9802955 IC50 = 41800 nM T09826 CQX6Y4 9837937 IC50 = 307000 nM T09826 CB1QT6 9851821 EC50 = 580 nM T09826 CW0TV4 9865348 IC50 = 640 nM T09826 C1R0GU 9865934 EC50 = 200 nM T09826 C71WVO 9887873 Ki = 400 nM T09826 CY4IG7 9889281 IC50 = 220 nM T09826 CLI8Z3 9898279 IC50 > 250000 nM T09826 CT2JF6 9907879 IC50 = 10000 nM T09826 CX13LY 9908423 IC50 = 20400 nM T09826 CKX02G 9909579 IC50 = 1400 nM T09826 CF0O4M 9918692 IC50 > 250000 nM T09826 CK67OG 9932270 IC50 = 130 nM T09826 C2RZE6 9953190 IC50 = 69 nM T09826 CNU9M5 9957793 IC50 = 300 nM T09826 CJ53PH 9975100 IC50 = 383 nM T09826 CBZ2D0 9979625 IC50 > 100000 nM T09826 CF0N4C 9980993 IC50 > 100000 nM T09826 C5S2ZX 9981804 IC50 = 1494 nM T09826 CO8T4X 9982858 IC50 = 220 nM T09826 CP0ZK9 9983085 IC50 = 11300 nM T09826 C9QV6A 10000564 IC50 = 5800 nM T09826 CKAU18 10001587 IC50 = 3200 nM T09826 CZ35OP 10006466 IC50 = 217 nM T09826 C42HFV 10023217 IC50 = 150 nM T09826 C8OE9R 10039843 IC50 = 129700 nM T09826 C1S6ZO 10053929 EC50 = 8 nM T09826 C5QWF2 10064551 IC50 < 10000 nM T09826 CA8HE1 10091894 IC50 = 4000 nM T09826 CY6K3R 10092735 IC50 = 167 nM T09826 CWQ1P3 10095286 IC50 = 24100 nM T09826 C0KU4D 10097407 IC50 = 180 nM T09826 CQ8X5W 10099547 IC50 > 625000 nM T09826 CSE5L1 10110293 IC50 = 2600 nM T09826 CK5Y9Q 10133241 IC50 = 38 nM T09826 CAL26K 10156768 IC50 = 140 nM T09826 COLS01 10177790 IC50 = 6400 nM T09826 C6C9KJ 10252111 IC50 = 1075 nM T09826 C12KCL 10271273 IC50 = 86 nM T09826 C2KP8J 10292113 IC50 = 300 nM T09826 CY53IN 10317270 IC50 = 4200 nM T09826 C5EYT8 10319267 IC50 = 190 nM T09826 C3K0SI 10321913 IC50 = 1331 nM T09826 C5FXU6 10323343 IC50 = 9328 nM T09826 CN0UE9 10346517 IC50 = 32000 nM T09826 C7RIC5 10362222 IC50 = 336 nM T09826 CTGD27 10363086 IC50 > 100000 nM T09826 C40KOF 10364204 IC50 = 1100 nM T09826 C93YBE 10366723 IC50 = 11 nM T09826 C9NZQ0 10366776 IC50 = 122 nM T09826 C7Q2UZ 10369338 IC50 = 2300 nM T09826 C67MHW 10386490 IC50 = 6600 nM T09826 CAN83B 10387283 IC50 = 19200 nM T09826 CPH0N9 10387840 IC50 = 1500 nM T09826 CLW5G1 10409273 IC50 > 100000 nM T09826 CS7YI3 10409274 IC50 = 3100 nM T09826 CJVI47 10411417 IC50 = 949 nM T09826 C8IU1M 10412775 IC50 = 700 nM T09826 CNZ9Q7 10433196 IC50 > 100000 nM T09826 CPK6J9 10439475 IC50 = 2602 nM T09826 CQTP21 10452851 IC50 = 143 nM T09826 CU1M0K 10453728 IC50 = 268 nM T09826 C6YPJ8 10453990 IC50 > 100000 nM T09826 C1MOR4 10455018 IC50 > 100000 nM T09826 C1F7EK 10455248 IC50 = 1500 nM T09826 CNB45M 10456398 IC50 = 29600 nM T09826 CFU75J 10460355 IC50 = 28 nM T09826 C26ESL 10482208 IC50 = 33 nM T09826 CJ0RE2 10485148 IC50 = 220000 nM T09826 CI6C1O 10506494 IC50 = 250 nM T09826 CYD7I0 10509674 IC50 = 4818 nM T09826 CIF7E4 10550144 IC50 = 1118 nM T09826 CULK80 10555744 IC50 = 120 ug.mL-1 T09826 CW56YA 10577898 IC50 = 190 nM T09826 CK63QR 10600972 IC50 = 200 nM T09826 CG2T5P 10626137 IC50 = 190 nM T09826 CU24QK 10676714 IC50 = 16618 nM T09826 CL4ZF6 10699214 IC50 = 2382 nM T09826 CLPH13 10745521 IC50 = 340 nM T09826 C26CVI 10768284 IC50 = 210 nM T09826 CX9F3O 10768720 IC50 = 520 nM T09826 CQ46NK 10769272 IC50 = 600 nM T09826 CXU9L1 10795337 IC50 = 2417 nM T09826 C8JWU1 10814294 IC50 = 160 nM T09826 CP56JD 10816483 IC50 = 100 nM T09826 CA2S8I 10933039 IC50 > 1000000 nM T09826 CU65BE 11317647 EC50 = 1950 nM T09826 CM6SF2 11414937 IC50 = 3000 nM T09826 CCG3Y1 11456414 IC50 = 120 ug.mL-1 T09826 CPQ3G6 11465894 EC50 = 1390 nM T09826 CQR90J 11623140 IC50 = 800000 nM T09826 CS80WY 11679800 IC50 > 250000 nM T09826 C92LND 11741224 IC50 = 232 nM T09826 CQ3E2J 11742279 IC50 = 1200 nM T09826 C9M7QD 11742280 IC50 > 100000 nM T09826 CEWF40 11743236 IC50 > 100000 nM T09826 C8A0NF 11755151 IC50 = 1113 nM T09826 CM76RE 11756340 IC50 = 1300 nM T09826 CNB5M3 11756382 IC50 = 1461 nM T09826 CER3U0 11788101 IC50 = 23800 nM T09826 C79UEW 11800135 IC50 = 140 nM T09826 CARZ73 11975877 IC50 = 6000 nM T09826 CD9Y6W 12304067 IC50 = 40000 nM T09826 CR7U6C 12632564 IC50 = 50000 nM T09826 CEC68V 12912322 IC50 > 250000 nM T09826 CK3MX1 12912363 IC50 > 250000 nM T09826 CR5UV0 13009345 EC50 = 17 nM T09826 CN3R8Q 13009346 EC50 = 100 nM T09826 CEW95R 13009351 EC50 = 30 nM T09826 C0DCE1 13009352 EC50 = 25 nM T09826 C53JGS 13009354 EC50 = 240 nM T09826 CU9G8A 13009355 EC50 = 130 nM T09826 CLE60O 13192381 EC50 = 450 nM T09826 C5LME0 13192383 EC50 = 4560 nM T09826 CJ5P3Y 13471631 IC50 = 4400 nM T09826 CR5C8E 13711981 IC50 = 21000 nM T09826 C6YX4Z 13714338 IC50 = 110630 nM T09826 CTI2K1 14083910 IC50 = 83140 nM T09826 CRHQ70 14194006 IC50 > 250000 nM T09826 C5P7AC 14194010 IC50 > 250000 nM T09826 CHD3G6 14203214 IC50 = 120000 nM T09826 CGLC61 14440698 IC50 = 9600 nM T09826 C9ED4C 14680465 IC50 = 1900 nM T09826 C23ANM 14804068 IC50 = 555000 nM T09826 CDKM67 14989978 IC50 = 150 nM T09826 C9FVU6 15589450 IC50 = 190 nM T09826 C4QMP2 16721067 IC50 = 42000 nM T09826 C3D7WE 17874201 EC50 = 700 nM T09826 CY6F1R 18336742 IC50 = 2000 nM T09826 C3AZJ2 19037238 EC50 = 270 nM T09826 C0EXH9 20089392 IC50 > 100000 nM T09826 C85AKW 20544405 IC50 > 100000 nM T09826 CUF9D8 20758666 EC50 = 1500 nM T09826 CUA6O7 20758668 EC50 = 500 nM T09826 CT8C5H 20758669 EC50 = 40 nM T09826 C3EHM4 21197160 EC50 = 3000 nM T09826 CDG36B 21350957 IC50 > 1000000 nM T09826 CGW4Q6 21580556 IC50 = 23800 nM T09826 C74HBW 21606527 IC50 = 110000 nM T09826 C69EDW 21636448 IC50 > 250000 nM T09826 C38TZQ 21918498 IC50 = 1500 nM T09826 C3KHM2 22569126 EC50 = 480 nM T09826 C3CW1K 22569130 EC50 = 750 nM T09826 C6CYN1 22569131 EC50 = 110 nM T09826 CQUR05 22569139 EC50 = 80 nM T09826 C6X8SE 22671105 EC50 = 51 nM T09826 CT54NE 22912790 IC50 = 30 nM T09826 CBU85X 23442826 EC50 = 240 nM T09826 C8L0KB 23662678 IC50 = 840 nM T09826 CMP12W 23662679 IC50 = 4300 nM T09826 C9GJD7 23666382 IC50 = 13000 nM T09826 CT3S9H 23666383 IC50 = 550 nM T09826 CV5AQ1 23705698 IC50 = 12000 nM T09826 CUPV08 24878308 IC50 = 370 nM T09826 CW4I9B 24878514 IC50 = 110 nM T09826 C1A9WX 24878522 IC50 = 160 nM T09826 CG02RD 24939224 IC50 = 6600 nM T09826 CK5V4T 24970451 IC50 = 23800 nM T09826 CQ7W8A 25067894 IC50 = 150000 nM T09826 C8GW1I 25241943 IC50 = 12800 nM T09826 C0D6VG 28392752 IC50 > 100000 nM T09826 CFO76L 42598162 IC50 = 8500 nM T09826 C9H1NM 42598163 IC50 = 11500 nM T09826 C89HEM 42598388 IC50 = 8200 nM T09826 CTW31D 44267388 IC50 = 42000 nM T09826 CZ67FA 44268667 IC50 = 1184 nM T09826 CP0BT5 44268675 IC50 = 505 nM T09826 C8PT0I 44273491 EC50 = 3500 nM T09826 CS6NT3 44273526 EC50 = 350 nM T09826 CG8H3R 44273527 EC50 > 10000 nM T09826 C7I1NX 44273528 EC50 = 250 nM T09826 C1WAE7 44273560 EC50 = 580 nM T09826 CQEW06 44273561 EC50 = 360 nM T09826 CUG08T 44273597 EC50 = 430 nM T09826 CIC13W 44273598 EC50 = 70 nM T09826 CC8W2J 44273599 EC50 = 300 nM T09826 CR1M9A 44273600 EC50 = 1200 nM T09826 CE6F2M 44273605 EC50 = 550 nM T09826 CBV2Y3 44273617 EC50 = 9500 nM T09826 CAK08Y 44273618 EC50 = 160 nM T09826 CT79EW 44273623 EC50 = 170 nM T09826 CZ6SM5 44273624 EC50 = 2800 nM T09826 CA8J9D 44273646 EC50 = 480 nM T09826 C8JWQ2 44273647 EC50 = 1000 nM T09826 CI72SY 44273652 EC50 = 90 nM T09826 CB0IL4 44273653 EC50 = 52 nM T09826 CA6LH1 44273654 EC50 = 1000 nM T09826 C8U2RI 44273699 EC50 = 270 nM T09826 CY9LQ3 44273700 EC50 = 580 nM T09826 C73SWH 44276082 IC50 = 500000 nM T09826 CJR6S0 44276312 IC50 = 400000 nM T09826 C4UMQ2 44283835 IC50 = 36000 nM T09826 CP1EH6 44290586 IC50 = 43200 nM T09826 C46LTQ 44290589 IC50 > 100000 nM T09826 C51OVA 44290590 IC50 > 100000 nM T09826 CCI29A 44290591 IC50 > 100000 nM T09826 C5PI6U 44290602 IC50 = 8600 nM T09826 C09JPK 44290621 IC50 = 1600 nM T09826 COS4W2 44290683 IC50 = 8200 nM T09826 CB7PQ0 44290711 IC50 = 16900 nM T09826 CA47LM 44290796 IC50 = 4700 nM T09826 C3PEZ2 44290797 IC50 = 11200 nM T09826 CTL54A 44290804 IC50 = 88000 nM T09826 C60SIM 44291373 IC50 > 100000 nM T09826 C4DE2F 44291412 IC50 = 34400 nM T09826 CF5AN3 44311920 IC50 = 3882 nM T09826 CA9YW3 44311921 IC50 = 4290 nM T09826 CIW8D1 44311922 IC50 = 11918 nM T09826 C8MC2H 44312069 IC50 = 1973 nM T09826 C9Y0AM 44312295 IC50 = 4842 nM T09826 C73YDG 44312296 IC50 = 4597 nM T09826 C4UA0D 44317168 IC50 = 43930 nM T09826 CB3A2R 44317204 IC50 = 30100 nM T09826 C90QNI 44317205 IC50 = 39000 nM T09826 CAQ25T 44317608 IC50 = 121830 nM T09826 C1MEF7 44324235 IC50 = 4000 nM T09826 C5CG8N 44324236 IC50 = 3800 nM T09826 CLT53Z 44324256 IC50 = 5500 nM T09826 C43NZU 44324259 IC50 = 2500 nM T09826 C4SEX7 44324261 IC50 = 260 nM T09826 C1D0QG 44324266 IC50 = 3200 nM T09826 C9FGW2 44324270 IC50 = 6800 nM T09826 C0RE5Y 44324306 IC50 > 30000 nM T09826 C76RXN 44324318 IC50 > 30000 nM T09826 C2XOY6 44324330 IC50 = 1000 nM T09826 C0H3ZI 44324343 IC50 = 1100 nM T09826 CW4QC1 44324446 IC50 = 470 nM T09826 C5KJ1F 44324457 IC50 = 3100 nM T09826 CLA40G 44324458 IC50 = 61 nM T09826 CKB5F3 44340622 EC50 = 650 nM T09826 C75BGC 44340751 EC50 = 1900 nM T09826 CQR38J 44340782 EC50 = 210 nM T09826 CA41TG 44340902 EC50 = 130 nM T09826 CCI2V3 44340903 EC50 = 55 nM T09826 CUMB62 44340904 EC50 = 210 nM T09826 C6UA8W 44340907 EC50 = 55 nM T09826 CX0VE8 44340908 EC50 = 37 nM T09826 CH38JI 44340930 EC50 = 160 nM T09826 CP52UL 44340931 EC50 = 510 nM T09826 CVU2G5 44340932 EC50 = 350 nM T09826 CWRA68 44340969 EC50 = 650 nM T09826 C89VOG 44340970 EC50 = 230 nM T09826 C96QBS 44340971 EC50 = 490 nM T09826 CC24ZH 44340972 EC50 = 570 nM T09826 CO6Z2E 44340973 EC50 = 1100 nM T09826 C8ADK3 44340974 EC50 = 90 nM T09826 CTR1H5 44355186 EC50 = 100 nM T09826 C1S7UQ 44355276 EC50 = 17 nM T09826 CJA3Y2 44355293 EC50 = 140 nM T09826 CM8QH9 44355294 EC50 = 80 nM T09826 C0JNW8 44355295 EC50 = 230 nM T09826 CGFJ50 44355298 EC50 = 32 nM T09826 C2T8XD 44355299 EC50 = 42 nM T09826 CC6A2E 44355300 EC50 = 20 nM T09826 C7US6F 44355330 EC50 = 26 nM T09826 CO2PA6 44355373 EC50 = 140 nM T09826 C01IZY 44355546 EC50 = 26 nM T09826 C1CF8Z 44355547 EC50 = 300 nM T09826 C6CF2D 44355564 EC50 = 40 nM T09826 C3AVL5 44373754 IC50 = 3600 nM T09826 CMF69S 44373774 IC50 = 69000 nM T09826 C8BM1Y 44373794 IC50 = 3500 nM T09826 CCR2I9 44374005 IC50 = 2200 nM T09826 CK2HJ6 44380928 IC50 = 6700 nM T09826 CE17VI 44380930 IC50 > 100000 nM T09826 CNV5B2 44381032 IC50 > 100000 nM T09826 C7WMZ4 44381291 IC50 = 31900 nM T09826 C4JXS9 44381325 IC50 = 3200 nM T09826 C37ESJ 44381326 IC50 > 100000 nM T09826 CTL57S 44382872 IC50 = 2100 nM T09826 C4OAQ6 44383179 IC50 = 1300 nM T09826 CNI31X 44383210 IC50 > 100000 nM T09826 CTN28X 44383263 IC50 > 100000 nM T09826 CAO3Y7 44383740 IC50 > 100000 nM T09826 C9AI7H 44383741 IC50 = 1800 nM T09826 C7CXJ0 44383814 IC50 = 1900 nM T09826 CI9KU2 44383861 IC50 > 100000 nM T09826 CUE0K3 44383864 IC50 > 100000 nM T09826 C7UK0Z 44384424 IC50 > 100000 nM T09826 CFY9O4 44384483 IC50 = 12100 nM T09826 C6XA3S 44395034 EC50 = 1000 nM T09826 CE3GQ1 44395040 EC50 = 160 nM T09826 C6C7IS 44395054 EC50 = 1040 nM T09826 C01RIL 44395078 EC50 = 150 nM T09826 CMD12L 44395100 EC50 = 1160 nM T09826 CA43GF 44395116 EC50 = 240 nM T09826 C1P0IC 44395196 EC50 = 190 nM T09826 C0L5KM 44399636 EC50 = 3000 nM T09826 CI67XZ 44399667 EC50 = 50 nM T09826 CT2V7J 44399668 EC50 = 70 nM T09826 CX25CW 44399679 IC50 = 4900 nM T09826 C0X6BK 44399697 EC50 = 420 nM T09826 CHV2L1 44399713 EC50 = 200 nM T09826 C5MEG7 44399714 EC50 = 410 nM T09826 C17RAS 44401260 IC50 = 392000 nM T09826 CWJL24 44401288 IC50 > 1000000 nM T09826 CR3JN2 44401681 IC50 = 250000 nM T09826 CXCM26 44401682 IC50 = 160000 nM T09826 CT4K5F 44401784 IC50 = 262000 nM T09826 CUB96N 44401847 IC50 = 960000 nM T09826 C90WTK 44401922 IC50 = 4000 nM T09826 CAC38H 44401925 IC50 = 630000 nM T09826 CXPJ93 44428908 IC50 = 59500 nM T09826 C2UQ1L 44428913 IC50 = 64300 nM T09826 CNT3L9 44454668 IC50 = 9000 nM T09826 CBC86V 44454669 IC50 = 8000 nM T09826 CIAB35 44479228 IC50 = 53700 nM T09826 C7UVA3 44565937 EC50 = 25 nM T09826 CYA0S4 44565938 EC50 = 38 nM T09826 C1KM4S 44565939 EC50 = 30 nM T09826 CXU6F8 44565940 EC50 = 30 nM T09826 C1QHV2 44565941 EC50 = 30 nM T09826 CH1GC9 44565942 EC50 = 23 nM T09826 CSOH56 44565943 EC50 = 22 nM T09826 C9B6MH 44565944 EC50 = 35 nM T09826 C5W3SL 44565945 EC50 = 17 nM T09826 CRD7M6 44565946 EC50 = 30 nM T09826 C3QCZ0 44565947 EC50 = 20 nM T09826 CQJ52K 44565949 EC50 = 800 nM T09826 CKT9Z5 44565950 EC50 > 3000 nM T09826 C7XBJ4 44565952 EC50 = 300 nM T09826 C8Y1PU 44565953 EC50 = 12 nM T09826 CU52EF 44565954 EC50 = 34 nM T09826 CU0GC6 44565955 EC50 = 20 nM T09826 CJHL69 44565956 EC50 = 22 nM T09826 CMAN06 44565957 EC50 = 16 nM T09826 CTUD59 44565958 EC50 = 3.3 nM T09826 C8XTY5 44565959 EC50 = 27 nM T09826 C2Q6DY 44565960 EC50 = 22 nM T09826 CJF6L9 44565961 EC50 = 19 nM T09826 CY9EA3 44565962 EC50 = 25 nM T09826 CGDZ65 44565963 EC50 = 35 nM T09826 CCE18F 44565964 EC50 = 30 nM T09826 C6IFZ9 44565965 EC50 = 29 nM T09826 C07XFL 44565966 EC50 = 31 nM T09826 C2L6MX 44584555 IC50 > 250000 nM T09826 C7JM8K 44604383 IC50 > 100000 nM T09826 C1PN9C 46224647 IC50 > 250000 nM T09826 CNC12E 46887586 IC50 > 250000 nM T09826 CQI2S5 46887678 IC50 > 250000 nM T09826 CPV4N6 46887679 IC50 > 250000 nM T09826 CR1JF6 46887680 IC50 > 250000 nM T09826 C6NPL9 46887682 IC50 > 250000 nM T09826 CN3KO1 46888244 IC50 > 250000 nM T09826 C4FOQ9 46888245 IC50 = 51800 nM T09826 C23BUR 46888246 IC50 > 250000 nM T09826 C10DYA 46888247 IC50 = 23800 nM T09826 CNF63K 46888248 IC50 > 250000 nM T09826 CX16CG 46888249 IC50 = 23800 nM T09826 C7Z8AK 46888250 IC50 > 250000 nM T09826 C6Z0OV 46888251 IC50 = 23800 nM T09826 CJEQ63 46888252 IC50 > 250000 nM T09826 CB36TZ 46888253 IC50 > 250000 nM T09826 C58XEI 46888254 IC50 > 250000 nM T09826 C1OMX0 46888255 IC50 > 250000 nM T09826 CUL8I2 46888256 IC50 > 250000 nM T09826 C3I1NG 46888257 IC50 > 250000 nM T09826 C8GOY7 46888258 IC50 = 23800 nM T09826 C38NOI 46888259 IC50 = 109300 nM T09826 CQP4R3 46888260 IC50 > 250000 nM T09826 CY6W1R 46888296 IC50 = 23800 nM T09826 C8NPJ6 46888298 IC50 = 23800 nM T09826 CJM78A 46888299 IC50 > 250000 nM T09826 C9O3GR 46888300 IC50 > 250000 nM T09826 CLN81T 46888301 IC50 > 250000 nM T09826 CQD47J 46888307 IC50 = 48600 nM T09826 CQ43PL 46888308 IC50 = 45100 nM T09826 CQ7H3G 46888311 IC50 > 250000 nM T09826 CR6TY2 46888312 IC50 > 250000 nM T09826 CR5SB4 46888313 IC50 = 131700 nM T09826 CK6YH8 46888320 IC50 > 250000 nM T09826 C4LXR1 46888321 IC50 > 250000 nM T09826 CLM5U7 46888322 IC50 > 250000 nM T09826 CTF0E5 46888323 IC50 > 250000 nM T09826 C06WJX 46888324 IC50 > 250000 nM T09826 CV1KB4 46914768 IC50 = 7200 nM T09826 C1FR4K 46914769 IC50 = 40000 nM T09826 CBX96T 46914770 IC50 = 16500 nM T09826 CFYS63 46914919 IC50 > 100000 nM T09826 CF28XZ 52921852 IC50 = 810 nM T09826 CP8F3H 52948084 IC50 = 13000 nM T09826 CEH2F9 53261771 EC50 = 27650 nM T09826 C6OC5F 54686375 IC50 = 10000 nM T09826 C45ETV 54736483 IC50 = 60000 nM T09826 C73QKP 57390614 IC50 = 180000 nM T09826 C37IJG 57397583 IC50 = 260000 nM T09826 CM7Q3S 57401109 IC50 = 250000 nM T09826 C1C0VM 58160590 IC50 = 25410 nM T09826 C5H6YW 70683609 EC50 > 3000 nM T09826 CQGK50 71459520 IC50 = 55000 nM T09826 C09XZN 85858741 IC50 = 10 ug.mL-1 T09826 CCOR96 86278368 EC50 = 563 nM T09826 CE2XU1 86280046 EC50 > 50000 nM T09826 CMA3L8 101600075 IC50 = 25000 nM T09826 C9U8ZQ 101653179 IC50 > 30000 nM T09826 CHK6Z0 117968363 IC50 > 50000 nM T09826 C30HXF 117968523 IC50 > 50000 nM T09826 C8MJS1 118737469 IC50 = 670 nM T09826 C6MK8B 122178582 IC50 > 50000 nM T09826 CG3P5S 122192375 EC50 > 100000 nM T09826 C1N5ZC 122192376 EC50 = 30340 nM T09826 CB5C1G 122192377 EC50 = 10080 nM T09826 C7EPG0 122192378 EC50 > 100000 nM T09826 CX3Y0R 122192379 EC50 > 100000 nM T09826 C9TM8V 122192380 EC50 > 100000 nM T09826 CY4EO0 122192381 EC50 > 100000 nM T09826 CZRS91 122192946 IC50 = 10000 nM T09826 C4DM8C 122491669 IC50 = 11240 nM T09826 C9X8KZ 132574430 IC50 = 42180 nM T09826 COE9R6 132574433 IC50 = 27390 nM T09826 C51AMJ 134130803 IC50 = 0.57 ug.mL-1 T09826 C6B7HM 134133214 IC50 = 22 ug.mL-1 T09826 C5V7BL 134133316 IC50 = 0.52 ug.mL-1 T09826 CQZ1J6 134135134 IC50 = 1.8 ug.mL-1 T09826 CI8VJ4 134135137 IC50 = 30 ug.mL-1 T09826 C3POG2 134135688 IC50 > 50000 nM T09826 C2O3NG 134136099 IC50 = 4.5 ug.mL-1 T09826 C5ABG9 134136339 IC50 = 5 ug.mL-1 T09826 C0AQS8 134136517 IC50 < 6 ug.mL-1 T09826 C3I0GC 134136603 IC50 = 15 ug.mL-1 T09826 CE9AS6 134136775 IC50 = 55 ug.mL-1 T09826 CBOX42 134138791 IC50 = 0.7 ug.mL-1 T09826 C3TU8P 134138793 IC50 = 17.5 ug.mL-1 T09826 C68JTQ 134139280 IC50 = 90 ug.mL-1 T09826 C8PEG1 134140951 IC50 = 2.4 ug.mL-1 T09826 CP8AI9 134142461 IC50 = 0.475 ug.mL-1 T09826 CH6MQ1 134142567 IC50 = 11 ug.mL-1 T09826 C9A1JY 134143508 IC50 = 12 ug.mL-1 T09826 CU5JO1 134143631 IC50 = 15 ug.mL-1 T09826 CMB30U 134144217 IC50 > 50000 nM T09826 CBJ18F 134145279 IC50 = 0.7 ug.mL-1 T09826 C3PF9N 134150635 IC50 = 50 ug.mL-1 T09826 CO6B8R 134150708 IC50 = 0.45 ug.mL-1 T09826 CBTJ76 134152787 IC50 = 31 ug.mL-1 T09826 C5SLA4 134153923 IC50 > 50000 nM T09826 C3HM9Q 134154564 IC50 = 12 ug.mL-1 T09826 CH4EN7 134155204 IC50 = 22 ug.mL-1 T09826 CWZ3Q9 134155778 IC50 = 4.4 ug.mL-1 T09826 CC9FM8 134156585 IC50 = 21 ug.mL-1 T09826 C47FCZ 134156695 IC50 = 0.7 ug.mL-1 T09826 C8ADP7 134156804 IC50 = 38 ug.mL-1 T09826 C3GCM7 134157712 IC50 > 50000 nM T09826 CGUM50 134157791 IC50 = 45 ug.mL-1 T09826 C57BSY 134589805 IC50 = 43700 nM T09826 COI3X8 134603858 IC50 = 15600 nM T09826 C4O1AN 134603859 IC50 = 25900 nM T09826 C41PKX 134603873 IC50 = 26000 nM T09826 C3L7ES 134603876 IC50 > 200000 nM T09826 C31WER 134603878 IC50 > 200000 nM T09826 CR8F5C 134603879 IC50 = 101000 nM T09826 CDH86P 134603881 IC50 = 33300 nM T09826 C6UH8R 134603884 IC50 = 60900 nM T09826 CZC7H3 134603886 IC50 = 154600 nM T09826 COVI15 134603888 IC50 = 91600 nM T09826 C5NR3V 134603904 IC50 = 72800 nM T09826 C47SQN 134603905 IC50 > 200000 nM T09826 CC7M9B 134603908 IC50 = 184200 nM T09826 C1DQY7 134603909 IC50 > 200000 nM T09826 CFJX62 134603912 IC50 = 71400 nM T09826 C7YCT8 134603913 IC50 = 92200 nM T09826 CL62NS 134603914 IC50 = 58600 nM T09826 CP76LG 134603916 IC50 = 35900 nM T09826 C0BXS2 134603917 IC50 = 82100 nM T09826 C1EQ6J 134603918 IC50 = 57700 nM T09826 CX08PD 134603928 IC50 > 200000 nM T09826 C8H7ZS 134603935 IC50 > 200000 nM T09826 CB4E2R 134603975 IC50 > 200000 nM T09826 C7T8WY 134603996 IC50 = 61200 nM T09826 COFI54 134603997 IC50 = 63600 nM T09826 CG8RJ9 135403790 IC50 = 870 nM T09826 CAOX53 135406264 IC50 = 900 nM T09826 C4NK0L 135407394 EC50 > 50000 nM T09826 CX86SO 135411729 EC50 > 50000 nM T09826 CT6M7E 135435051 IC50 > 200000 nM T09826 CUO4X6 135437964 IC50 = 71 nM T09826 C3YH2A 135492582 IC50 = 170 nM T09826 CNSO96 135871337 IC50 = 3760 nM T09826 C45EIW 135939142 IC50 = 7400 nM T09826 CU67OL 135939143 IC50 > 100000 nM T09826 C75HEQ 135939144 IC50 > 100000 nM T09826 C86FAY 135939145 IC50 > 100000 nM T09826 C6MAG4 136726274 EC50 > 50000 nM T09826 CZM2N8 137289827 IC50 = 15 ug.mL-1 T09826 C36PSK 137638477 EC50 = 63430 nM T09826 CG5M4F 137645246 EC50 > 50000 nM T09826 C2BJ1A 137646923 EC50 = 1226 nM T09826 CRH4A0 137648926 EC50 > 50000 nM T09826 CJ0LG4 137658592 EC50 = 381 nM T09826 C9ME4X 137659985 IC50 > 50000 nM T09826 C35TXH 138377597 IC50 = 29 nM T09826 C96FIT 142372764 IC50 = 88300 nM T09826 CIJ78Z 145950337 IC50 = 72680 nM T09826 CD56IQ 145950672 IC50 = 82080 nM T09826 CM9XH4 145952636 IC50 = 83250 nM T09826 C9NBC5 145953065 IC50 = 70610 nM T09826 C16ETI 145954110 IC50 = 82030 nM T09826 CMPX68 145955703 IC50 = 73110 nM T09826 COZ6S1 145956088 IC50 = 50930 nM T09826 C20LCF 145959577 IC50 = 72770 nM T09826 CJ7X9K 145972200 IC50 = 67530 nM T09826 C8EG5Q 145973453 IC50 = 84560 nM T09826 C3RWK4 145974823 IC50 = 43850 nM T09826 COIT57 145977875 IC50 = 44790 nM T09826 COZ0U7 146433455 IC50 = 200000 nM T09826 C2L4BQ 146433456 IC50 > 200000 nM T09826 CCT4Z3 146433460 IC50 = 167600 nM T09826 CR5NS8 146433531 IC50 = 100400 nM T09826 CZ6T8I 146433532 IC50 = 58300 nM T09826 C8K3YV 146433533 IC50 = 61000 nM T09826 CF3TQ8 146433534 IC50 = 103900 nM T09826 CVT82N 146433594 IC50 > 200000 nM T09826 CY3M7A 146433600 IC50 = 187400 nM T09826 CVI5Z7 146433615 IC50 = 178400 nM T09826 CA1RQ4 147522895 IC50 > 10000 nM T09826 C4SR8E 148471279 IC50 > 10000 nM T09826 C3VH2Q 151325855 IC50 = 1054 nM T09826 CB82LR 151546137 IC50 > 10000 nM T09826 CQ7OJ5 152715282 IC50 > 10000 nM T09826 C0PVM6 153370104 IC50 > 10000 nM T09826 C32YUG 153370108 IC50 > 10000 nM T09826 CFJ12N 153370109 IC50 > 10000 nM T09826 CW0OM8 153370112 IC50 > 10000 nM T09826 CO4D3Q 153370113 IC50 = 3750 nM T09826 C6AUZ0 153370116 IC50 > 10000 nM T09826 C1JN2H 153370118 IC50 > 10000 nM T09826 C80LZF 153370124 IC50 > 10000 nM T09826 CSM80A 153370126 IC50 > 10000 nM T09826 C72LJX 153370129 IC50 > 10000 nM T09826 C2IAT1 153370141 IC50 = 2360 nM T09826 CO73HF 153370142 IC50 > 10000 nM T09826 CV5TU1 153370145 IC50 > 10000 nM T09826 C0RB7T 153455863 IC50 = 172500 nM T09826 CFBM09 155515657 IC50 > 10000 nM T09826 C97UAV 155517975 IC50 > 10000 nM T09826 C32QTC 155518845 IC50 = 69650 nM T09826 C1Q2FH 155520735 IC50 = 34800 nM T09826 CEF41K 155521372 IC50 = 61000 nM T09826 C29VST 155529673 IC50 = 1790 nM T09826 C0PQ9F 155531850 IC50 > 10000 nM T09826 CVB45T 155532863 IC50 > 10000 nM T09826 CMPL28 155546084 IC50 = 63600 nM T09826 CN28RI 155550639 IC50 = 31300 nM T09826 C6W3HF 155555769 IC50 > 200000 nM T09826 CK3U9T 155557567 IC50 > 10000 nM T09826 C83GLA 155567561 IC50 = 69600 nM T09826 D00DXV 9895647 IC50 = 120 ug.mL-1 T09826 D01BKS 9918693 IC50 > 250000 nM T09826 D01QKX 44567153 IC50 = 900 nM T09826 D03SPJ 73568 IC50 = 40000 nM T09826 D05ZVR 4461 IC50 = 62000 nM T09826 D07ILP 97226 IC50 = 110 nM T09826 D0A4EA 445639 IC50 = 31000 nM T09826 D0BS6Q 3115 IC50 = 2700 nM T09826 D0E8ZH 2392 IC50 = 22860 nM T09826 D0G2JZ 1464 IC50 > 50000 nM T09826 D0J5OV 442674 IC50 = 50 nM T09826 D0L8BN 44559995 IC50 = 29000 nM T09826 D0RL8X 9981577 IC50 = 2300 nM T09826 D0T3PW 5281672 IC50 = 11.9 ug.mL-1 T32262 D00MXN 25019940 Ki = 0.021 nM T32262 D0G5ME 11319053 Ki = 0.77 nM T32262 D0IA9Y 53472683 Ki = 0.023 nM T32262 D0L5GH 6918509 Ki = 0.01 nM T32262 D0V9VG 51049968 Ki = 0.027 nM T32262 CW2XB1 9978597 Ki = 78 nM T32262 CSY53V 10077700 Ki = 0.012 nM T32262 C9RXY3 10102983 IC50 = 146 nM T32262 CEP07A 10340395 Ki = 280 nM T32262 CC36IR 10340456 Ki = 309 nM T32262 C0EQX7 10394458 Ki = 0.011 nM T32262 C01PKW 10416497 IC50 = 0.074 nM T32262 C0YSQ7 10416713 Ki = 0.005 nM T32262 C4S2JZ 10433192 IC50 = 5500 nM T32262 C69MPT 10438558 IC50 = 3.2 nM T32262 CS94QC 10453991 Ki = 607 nM T32262 CXP35B 10483468 IC50 = 87 nM T32262 CHNT90 10483685 Ki = 32 nM T32262 CFG4O3 11156698 IC50 = 4.4 nM T32262 CSQP28 11157609 Ki = 6900 nM T32262 CFC0L9 11157626 IC50 = 224 nM T32262 C1R4CH 11158071 Ki = 0.22 nM T32262 C0KY1X 11168000 Ki = 11 nM T32262 C8BLU1 11169408 IC50 = 1.9 nM T32262 C6Q9MF 11169454 IC50 = 0.34 nM T32262 C1TY6Q 11180666 Ki = 1.7 nM T32262 CR4O1G 11191890 IC50 = 10 nM T32262 CXF10W 11192602 Ki = 0.5 nM T32262 CV6NF8 11192748 IC50 = 1.3 nM T32262 CKE6B8 11204498 IC50 = 0.19 nM T32262 CTS40R 11204595 Ki = 0.039 nM T32262 CQI1R0 11215322 Ki = 427 nM T32262 CNL48A 11215412 IC50 = 12 nM T32262 CJ39MV 11215446 IC50 = 0.49 nM T32262 CA7H8W 11215502 Ki = 983 nM T32262 CNW94U 11215639 Ki = 6400 nM T32262 C6BZ8W 11225752 Ki = 2.7 nM T32262 C2U7FL 11226747 IC50 = 1.4 nM T32262 CAY0X1 11227287 Ki > 10000 nM T32262 C2I7CU 11238250 IC50 = 28 nM T32262 CJD59I 11238677 IC50 = 0.42 nM T32262 C7GZ9Q 11238717 Ki = 2800 nM T32262 CSZ2M3 11249157 IC50 = 30 nM T32262 C7J4WT 11250445 IC50 = 0.63 nM T32262 CMX8H7 11250446 IC50 = 0.98 nM T32262 CT2KR7 11261842 Ki = 965 nM T32262 C39NJZ 11273798 IC50 = 4.8 nM T32262 C1I4RB 11284233 Ki = 0.9 nM T32262 CL41QP 11286085 IC50 = 776.25 nM T32262 CF65RC 11295168 IC50 = 3.1 nM T32262 CGPS72 11295951 IC50 = 0.46 nM T32262 C3HZ9A 11297807 IC50 = 588.84 nM T32262 CHM45S 11308069 IC50 = 0.099 nM T32262 CKQ01L 11308219 IC50 = 0.089 nM T32262 CXF31N 11330650 Ki = 685 nM T32262 CGML40 11330786 Ki = 320 nM T32262 C6TFR2 11341430 IC50 = 3.8 nM T32262 CAV4B2 11341642 IC50 = 0.94 nM T32262 CR9J6K 11342207 Ki = 853 nM T32262 CKTZ78 11351794 Ki = 22 nM T32262 C2SN5F 11354531 Ki = 0.14 nM T32262 C7L3VT 11364682 IC50 = 0.21 nM T32262 CPV21T 11364735 Ki = 0.3 nM T32262 C89EDQ 11365194 IC50 = 1583 nM T32262 CR6H4L 11375693 Ki = 2.4 nM T32262 CM87TN 11375696 IC50 = 120 nM T32262 C18WDP 11377534 Ki = 0.023 nM T32262 CR2F7Y 11387141 IC50 = 2.1 nM T32262 CJ7U4X 11387595 Ki = 0.9 nM T32262 CGY80S 11388586 Ki = 0.055 nM T32262 C4YTL3 11397560 Ki = 3.6 nM T32262 CJ7B1C 11398863 IC50 = 4.8 nM T32262 CZQ35I 11409395 IC50 = 97 nM T32262 CB6TC2 11410749 IC50 = 34 nM T32262 CJ1CM9 11411030 IC50 = 0.39 nM T32262 CTV17E 11421827 Ki = 22 nM T32262 C54GDM 11422298 IC50 = 0.078 nM T32262 CZU3S7 11423175 IC50 = 4466.84 nM T32262 C0YT2F 11432183 IC50 = 8.6 nM T32262 CHGT51 11432505 Ki = 10 nM T32262 C6CE9W 11432931 Ki = 0.7 nM T32262 CYZ92S 11434781 IC50 = 707.95 nM T32262 C3B2TE 11443894 IC50 = 35 nM T32262 C56IND 11444574 IC50 = 7.4 nM T32262 CRE9W2 11444589 Ki = 156 nM T32262 CAI0X1 11444699 Ki = 6100 nM T32262 C62PUD 11445240 Ki = 0.28 nM T32262 C6CD1Y 11453687 Ki = 83 nM T32262 C2MOP7 11454113 Ki = 51 nM T32262 CW5BO3 11456078 IC50 = 1.6 nM T32262 CJU06L 11456102 Ki = 295 nM T32262 CH6S7Z 11456201 IC50 = 0.88 nM T32262 C1U8CX 11466363 IC50 = 1.5 nM T32262 CY1EG6 11467108 IC50 = 1 nM T32262 C16NBP 11467753 Ki = 0.0073 nM T32262 CFOC05 11478841 IC50 = 0.83 nM T32262 CFC93K 11478962 IC50 = 0.13 nM T32262 CHF3T7 11495985 IC50 = 495 nM T32262 C9WD3C 11497403 Ki = 855 nM T32262 C0P1QE 11498219 IC50 = 0.02 nM T32262 CN2Y7Z 11505361 Ki = 2000 nM T32262 C01MDL 11512851 IC50 = 0.063 nM T32262 CQUV12 11512928 Ki = 1.1 nM T32262 CV92TG 11513230 IC50 > 300000 nM T32262 C4D0FS 11519899 Ki = 110 nM T32262 CT97KM 11520007 Ki = 0.63 nM T32262 CFDQ43 11520022 Ki = 339 nM T32262 C8EI9U 11520204 IC50 = 0.057 nM T32262 CDG8W2 11526993 Ki = 3.5 nM T32262 C5TFH3 11527287 Ki = 720 nM T32262 CU8CE9 11532845 Ki = 96 nM T32262 CHF2N8 11534977 IC50 = 17000 nM T32262 CAD16K 11541560 Ki = 1.1 nM T32262 CJ6E4C 11541725 Ki = 27 nM T32262 CHS87Q 11548734 IC50 = 23 nM T32262 C7SK0A 11549001 IC50 = 450 nM T32262 C9HT8K 11549159 IC50 = 0.022 nM T32262 CR79TM 11555955 Ki = 46 nM T32262 CEK1F3 11562434 Ki = 3.7 nM T32262 C8DIQ5 11570464 Ki = 5337 nM T32262 C20RJY 11570753 Ki = 1050 nM T32262 CE4IT9 11571094 Ki = 19 nM T32262 CP8M4A 11576078 Ki = 270 nM T32262 CA9TQ4 11578671 IC50 = 17000 nM T32262 C18FPK 11584808 Ki = 1.7 nM T32262 C9LQD0 11585317 Ki = 6.3 nM T32262 CG4FL3 11592648 IC50 = 0.068 nM T32262 CCAQ30 11599135 IC50 = 1.8 nM T32262 C4O7JT 11599531 IC50 = 120 nM T32262 C4X7NH 11599798 IC50 = 0.053 nM T32262 C30LBG 11599872 IC50 = 0.13 nM T32262 CO0V9M 11599913 IC50 = 0.011 nM T32262 CNU10O 11606400 Ki = 0.69 nM T32262 CBV9D3 11621504 IC50 = 0.01 nM T32262 CNT8V6 11628731 Ki = 11 nM T32262 C7Z4AE 11636224 IC50 > 300000 nM T32262 CWE5X4 11650307 IC50 = 193 nM T32262 CK3UO8 11657395 IC50 = 0.044 nM T32262 C08UGA 11671386 Ki = 2900 nM T32262 C9B6GR 11678239 Ki = 3.2 nM T32262 CO4DL5 11678456 Ki = 20000 nM T32262 C1JFI5 11685954 IC50 = 0.017 nM T32262 CX4Q2U 11691938 Ki = 3.1 nM T32262 C69HMB 11692140 Ki = 4 nM T32262 C87ZSQ 11692206 Ki = 583 nM T32262 CO3EI9 11692628 Ki = 1.1 nM T32262 C4XFK0 11693761 IC50 = 44 nM T32262 C29VOY 11699891 Ki = 3.9 nM T32262 CVLK50 11706251 Ki = 46 nM T32262 CG0B5Q 11706981 Ki = 0.07 nM T32262 C8RCQ9 11707040 Ki = 11 nM T32262 C7XJ8D 11713729 Ki = 575 nM T32262 C2NC5F 11713849 Ki = 1249 nM T32262 CF76KX 11721278 Ki = 1.1 nM T32262 CW8V7S 11752904 Ki = 1.4 nM T32262 C24ODM 11753021 Ki = 1.4 nM T32262 CX19UV 11753024 IC50 = 6 nM T32262 C1EMS2 11785573 IC50 = 4.8 nM T32262 CB17JY 11785754 IC50 = 12 nM T32262 C01QPC 11786529 Ki = 51 nM T32262 CE0HF8 11786642 IC50 = 0.38 nM T32262 C5RPV6 11848645 Ki = 220 nM T32262 CY6X8K 11848646 Ki = 43 nM T32262 C81SEQ 11848647 Ki = 270 nM T32262 C1PN7A 11848698 Ki = 9000 nM T32262 C0NF3B 11848750 Ki = 75 nM T32262 CHL78I 11848753 Ki = 1750 nM T32262 CL4S1Z 11848755 Ki = 495 nM T32262 C7KZL1 11848798 Ki = 1900 nM T32262 C9EAL0 11848800 Ki = 228 nM T32262 CPSU54 11848855 Ki = 74 nM T32262 CNP83T 11848857 Ki = 695 nM T32262 CWRO47 11848908 Ki = 41 nM T32262 C23ZVT 11848963 Ki = 170 nM T32262 C67WMH 11848964 Ki = 95 nM T32262 C8K9IP 11848965 Ki = 54 nM T32262 C9E7VN 11848966 Ki = 42 nM T32262 CHM18G 11848968 Ki = 105 nM T32262 C4ZY7K 11849020 Ki = 96 nM T32262 C4VI7D 11849023 Ki = 635 nM T32262 CS17WY 11849024 Ki = 205 nM T32262 C1LYJ0 11849025 Ki = 17 nM T32262 C21UVM 11849147 Ki = 80 nM T32262 CUT84W 16115156 IC50 = 107.15 nM T32262 C2I4RM 16745090 Ki = 185 nM T32262 CR79HP 21102037 IC50 = 2 nM T32262 CK10IC 21102038 IC50 = 3.7 nM T32262 CZ1Q0N 21102224 EC50 = 31 nM T32262 C9FW6Z 23627980 Ki = 35 nM T32262 CLQ2B0 23654987 Ki = 0.3 nM T32262 CAH83C 23656586 Ki = 4400 nM T32262 CE4ZM7 23656587 Ki = 770 nM T32262 CYKB10 23656588 Ki = 9900 nM T32262 CWMD21 23656749 Ki = 470 nM T32262 CBS03U 23656750 Ki = 1700 nM T32262 CRET24 23656751 Ki = 1100 nM T32262 CGR12U 23656752 Ki = 470 nM T32262 CCE3B5 23656753 Ki = 610 nM T32262 C7CO2B 23656918 Ki = 37 nM T32262 C3JIP1 23656919 Ki = 93 nM T32262 CDL81I 23656920 Ki = 4.2 nM T32262 CRQ31C 23656921 Ki = 0.19 nM T32262 CV96FP 23656922 Ki = 4.9 nM T32262 CM27YU 23657089 Ki = 0.5 nM T32262 CH2L9G 24756611 EC50 = 12 nM T32262 CVG14A 24756612 EC50 = 130 nM T32262 C7DL3K 24756690 IC50 = 0.33 nM T32262 CF3J6T 24756767 IC50 = 5.9 nM T32262 CF40KL 24756768 IC50 = 34 nM T32262 CQ3X4L 24756769 IC50 = 15 nM T32262 C3X4NK 24756770 IC50 = 460 nM T32262 C08WIS 24853163 Ki = 88 nM T32262 CZK38U 24853164 Ki = 2 nM T32262 CJ4T7O 24853374 Ki = 32 nM T32262 CO73CZ 24862842 Ki = 68 nM T32262 C0UN7H 24863246 Ki = 28 nM T32262 C84JXU 24863323 Ki = 0.55 nM T32262 CUY1O2 24863332 Ki = 0.27 nM T32262 CV29XP 24863333 Ki = 0.23 nM T32262 CJIN21 24863334 Ki = 0.65 nM T32262 CAFZ85 25019993 Ki = 0.034 nM T32262 C0X8DC 25034109 Ki = 0.55 nM T32262 CY8EP0 25110584 Ki = 6.31 nM T32262 CURE82 25151777 Ki = 3.981 nM T32262 CSP1W0 25151968 Ki = 3.162 nM T32262 CUM6S8 25152167 Ki = 5.012 nM T32262 C78MVE 25152169 Ki = 2.512 nM T32262 CYR8F9 25152367 Ki = 7.943 nM T32262 CP0U4K 25152370 Ki = 12.59 nM T32262 CWI75J 25152560 Ki = 15.85 nM T32262 CN8BM0 25152561 Ki = 25.12 nM T32262 C2OB9H 25152563 Ki = 125.89 nM T32262 CP0W7T 25152564 Ki = 125.89 nM T32262 C3ZWB2 25152765 Ki = 6.31 nM T32262 C0EL1C 25152766 Ki = 3.981 nM T32262 C2K3LX 25152981 Ki = 50.12 nM T32262 C3BI5L 25152984 Ki = 25.12 nM T32262 CA64HU 25152985 Ki = 25.12 nM T32262 C8LK9M 25153832 Ki = 1.585 nM T32262 C9TA6K 25154032 Ki = 3.981 nM T32262 C9MW8O 25154034 Ki = 2.512 nM T32262 C2KTS7 25181509 Ki = 0.039 nM T32262 CIM67A 25227362 Ki = 0.51 nM T32262 CHRS21 44273362 IC50 = 70000 nM T32262 CM4PQ5 44273364 IC50 = 51000 nM T32262 CVSZ14 44273516 IC50 > 100000 nM T32262 CDX27H 44273596 IC50 = 8550 nM T32262 CS53AM 44273608 IC50 = 5000 nM T32262 C3S5NZ 44273609 IC50 = 95000 nM T32262 C24FZC 44273610 IC50 = 7000 nM T32262 CP48DY 44273621 IC50 = 6900 nM T32262 C83HLE 44273622 IC50 = 4275 nM T32262 CDU4K9 44273716 IC50 > 3000 nM T32262 CTO2F1 44273717 IC50 > 3000 nM T32262 C93UJI 44273718 IC50 = 220 nM T32262 CIP61B 44273804 IC50 = 3000 nM T32262 CC02NK 44273825 IC50 = 10000 nM T32262 CCG57H 44273826 IC50 = 10000 nM T32262 C2K8FX 44273827 IC50 = 10000 nM T32262 C3BYF4 44273842 IC50 = 45000 nM T32262 C20HDP 44273843 IC50 > 100000 nM T32262 CIX61G 44273844 IC50 = 200 nM T32262 CIE3V4 44273845 IC50 > 10000 nM T32262 CHB1T0 44273857 IC50 = 360 nM T32262 C1E0JP 44273858 IC50 = 470 nM T32262 C12THF 44273867 IC50 = 9000 nM T32262 CVE0I8 44273868 IC50 = 300 nM T32262 CS2EI3 44273869 IC50 = 8000 nM T32262 C6DU4X 44273870 IC50 = 24000 nM T32262 CIU4V7 44273871 IC50 = 10000 nM T32262 C1AP7W 44273878 IC50 = 1200 nM T32262 C9Z1IG 44273880 IC50 = 2700 nM T32262 CJG5M9 44273881 IC50 = 6500 nM T32262 CB8NE4 44273909 IC50 = 4000 nM T32262 C4BUD5 44273948 IC50 > 10000 nM T32262 CNRA07 44273949 IC50 = 3400 nM T32262 CBCP21 44273950 IC50 = 32000 nM T32262 C7X1FO 44273967 IC50 = 24000 nM T32262 CAO4P7 44273969 IC50 > 100000 nM T32262 CD7J9B 44273976 IC50 = 490 nM T32262 C0ZBP1 44273979 IC50 = 280 nM T32262 CA02ZL 44273980 IC50 > 10000 nM T32262 CR54UE 44273987 IC50 = 18000 nM T32262 CVM9S8 44273992 IC50 = 80000 nM T32262 CQE3U0 44273994 IC50 = 4790 nM T32262 C36GES 44274008 IC50 = 10000 nM T32262 C6JCG2 44274013 IC50 > 10000 nM T32262 CG0A2V 44274014 IC50 = 4500 nM T32262 CXCT49 44274025 IC50 = 620 nM T32262 C02GLR 44274032 IC50 = 205 nM T32262 CO60FW 44274035 IC50 = 10000 nM T32262 C93URN 44274036 IC50 = 10000 nM T32262 CQ5O3Z 44274037 IC50 = 14000 nM T32262 CV3A8Z 44274039 IC50 > 10000 nM T32262 C0WQV6 44274073 IC50 = 10000 nM T32262 CGJ56K 44274074 IC50 > 100000 nM T32262 C6Z9AJ 44274076 IC50 > 100000 nM T32262 C5Y7LE 44274096 IC50 > 3000 nM T32262 CV17HE 44274097 IC50 > 10000 nM T32262 CNO3Y6 44274098 IC50 = 170 nM T32262 C98IRQ 44274099 IC50 = 4500 nM T32262 CXVF03 44274101 IC50 = 3000 nM T32262 CBYZ92 44323001 IC50 = 17000 nM T32262 CG2WX7 44323086 IC50 > 100000 nM T32262 C0KZ2L 44323087 IC50 > 100000 nM T32262 C0Q6DS 44323095 IC50 = 5200 nM T32262 C6G1KZ 44323097 IC50 = 12000 nM T32262 C64YGA 44323110 IC50 = 96000 nM T32262 CD2S7Q 44323139 IC50 = 33000 nM T32262 CIO08E 44323180 IC50 = 9900 nM T32262 CC4YF1 44323332 IC50 = 41000 nM T32262 CFAY53 44323338 IC50 = 37000 nM T32262 C12WJT 44323339 IC50 > 100000 nM T32262 C5OGN1 44323341 IC50 = 74000 nM T32262 C49QHD 44403853 IC50 = 13000 nM T32262 C4TF8U 44403854 IC50 = 1000 nM T32262 C3AU1P 44403855 IC50 = 200 nM T32262 CZJ63F 44403856 IC50 = 226 nM T32262 CWS0U9 44403857 IC50 = 250 nM T32262 C1LW2J 44403858 IC50 = 44 nM T32262 C3X7GN 44403859 IC50 = 4.7 nM T32262 CJK6A8 44403860 IC50 = 0.2 nM T32262 CU3C1O 44403861 IC50 = 0.03 nM T32262 CNR30J 44403862 IC50 = 0.05 nM T32262 CJ6PA5 44403914 IC50 = 50000 nM T32262 C15ZXC 44403915 IC50 > 300000 nM T32262 CF24BX 44403916 IC50 > 300000 nM T32262 CUDT41 44403917 IC50 = 10300 nM T32262 CSA8I5 44403918 IC50 = 196000 nM T32262 CIR8W1 44404069 IC50 = 40000 nM T32262 CJ69ZX 44416436 IC50 = 373 nM T32262 C9X3NK 44416437 Ki = 143 nM T32262 CWYX41 44416442 Ki = 1000 nM T32262 C0GQL1 44416488 Ki = 3800 nM T32262 C2UHG0 44416512 IC50 = 715 nM T32262 C7JI1G 44416513 Ki = 1055 nM T32262 C1ZM4Q 44416514 IC50 = 220 nM T32262 C5HIN3 44416516 Ki = 20000 nM T32262 CXY19R 44416912 Ki = 11 nM T32262 CDS7E4 44417049 Ki = 104 nM T32262 CODP98 44417050 Ki = 27 nM T32262 CQO2U8 44420227 Ki = 87 nM T32262 CAM5F1 44420228 Ki = 38 nM T32262 C5LB7G 44420231 Ki = 29 nM T32262 CY2F3Q 44420235 Ki = 20 nM T32262 C46VUS 44420236 Ki = 8.7 nM T32262 CC9MN0 44420240 Ki = 20 nM T32262 CM89QF 44420241 Ki = 6.8 nM T32262 C4V5SX 44420245 Ki = 15 nM T32262 CO9BH3 44420250 Ki = 10 nM T32262 C7ANU1 44420255 Ki = 25 nM T32262 C8TE2M 44420256 Ki = 12 nM T32262 CL2FN9 44420260 Ki = 9.5 nM T32262 CFWC52 44420261 Ki = 17 nM T32262 C1T6IE 44420286 Ki = 103 nM T32262 CFPY38 44420287 Ki = 48 nM T32262 C3NQT1 44420290 Ki = 1050 nM T32262 CZY17T 44420691 IC50 = 380.19 nM T32262 C3H1EF 44420692 IC50 = 67.61 nM T32262 CWX81Y 44420693 IC50 = 5754.4 nM T32262 CZS90I 44421021 EC50 = 0.2 nM T32262 C0NAY5 44454954 Ki = 390 nM T32262 CLV3J4 44455041 Ki = 166 nM T32262 CPS61E 44455043 Ki = 155 nM T32262 CY4N5D 44455078 Ki = 213 nM T32262 CY7OU8 44455080 Ki = 71 nM T32262 CECP81 44455153 Ki = 42 nM T32262 CJQ05D 44455188 Ki = 2050 nM T32262 CJ81LT 44455348 Ki = 3400 nM T32262 CXUZ08 44455457 Ki = 140 nM T32262 CB5T0Z 44468576 Ki = 0.094 nM T32262 C9C1RH 44468711 Ki = 0.5 nM T32262 CS2AV5 44469523 Ki = 0.11 nM T32262 C91APQ 44469664 Ki = 0.019 nM T32262 C31OVU 44469946 Ki = 0.021 nM T32262 C63BGP 44470090 Ki = 0.045 nM T32262 CVR8Q5 44562895 Ki = 5.5 nM T32262 CMRN61 44562896 Ki = 41 nM T32262 CYR7O0 44562897 Ki = 13 nM T32262 C9J2TE 44562936 Ki = 32 nM T32262 CG6A2F 44562937 Ki = 26 nM T32262 C2JZI8 44562938 Ki = 100 nM T32262 C35UFM 44562939 Ki = 15 nM T32262 CMI43S 44562982 Ki = 18 nM T32262 CZ2IV8 44562983 Ki = 62 nM T32262 C7XS9M 44562984 Ki = 23 nM T32262 CKA21W 44562985 Ki = 9.5 nM T32262 CQ8NJ3 44563025 Ki = 15 nM T32262 CPE7L6 44563026 Ki = 120 nM T32262 C8BMF5 44563027 Ki = 250 nM T32262 CV8BX9 44563028 Ki = 2.7 nM T32262 CFS8T3 44563050 Ki = 2.1 nM T32262 C5GLD7 44563051 Ki = 21 nM T32262 C0MX4G 44563052 Ki = 1.9 nM T32262 C4USA7 44563089 Ki = 26 nM T32262 CYCA43 44563090 Ki = 4.3 nM T32262 CAY83X 44563091 Ki = 37 nM T32262 C02GYS 44563123 Ki = 22 nM T32262 CQ1GS6 44563124 Ki = 31 nM T32262 C7RF8D 44563125 Ki = 36 nM T32262 CX10VW 44563126 Ki = 13 nM T32262 C8NI7J 44563160 Ki = 9.6 nM T32262 CP9KF1 44563161 Ki = 7.1 nM T32262 CE68LK 44563162 Ki = 4.7 nM T32262 C4XLF1 44563200 Ki = 2.2 nM T32262 CBN70V 44570375 Ki = 230 nM T32262 CN08BL 44570421 Ki = 2700 nM T32262 C8WAM1 44570422 Ki = 34 nM T32262 CU79ER 44570461 Ki = 130 nM T32262 CO7Q6R 44570462 Ki = 2600 nM T32262 CF5U3J 44570463 Ki = 520 nM T32262 CV07RL 44570498 IC50 = 10 nM T32262 CS0P9O 44570499 Ki = 13 nM T32262 CN82WG 44570536 Ki = 35 nM T32262 CKN09A 44570578 Ki = 2.3 nM T32262 C3P8KA 44570579 Ki = 0.61 nM T32262 C9U7GK 44570580 Ki = 1.2 nM T32262 C0AL8Y 44570614 Ki = 0.87 nM T32262 CH4ZR3 44570615 Ki = 1.7 nM T32262 CUT6X5 44570616 Ki = 0.21 nM T32262 C38SLX 44583379 IC50 = 0.18 nM T32262 CRJ69Y 44593445 Ki = 1.7 nM T32262 CVKF91 44593545 Ki = 0.23 nM T32262 CH32KB 45267476 Ki = 0.12 nM T32262 C6BC5R 45267481 Ki = 0.28 nM T32262 C9CFX4 45269221 Ki = 2.2 nM T32262 C2S5JO 45271740 Ki = 1.4 nM T32262 CPUN79 45271754 Ki = 1.1 nM T32262 CBCA26 45273525 Ki = 9.7 nM T32262 CIPX17 45485590 Ki = 45 nM T32262 CI10RQ 45485600 Ki = 23 nM T32262 CDP21J 45485605 Ki = 0.13 nM T32262 CPVU61 45485609 Ki = 25 nM T32262 C6IG2K 45485621 Ki = 800 nM T32262 C58VXQ 45485625 Ki = 1.9 nM T32262 CF7Y8H 45485631 Ki = 14 nM T32262 CMI83V 45485640 Ki = 0.55 nM T32262 CP87FU 45485645 Ki = 1.6 nM T32262 CLJF04 45485646 Ki = 1.2 nM T32262 CQE7Z0 45485654 Ki = 3.7 nM T32262 C5J4CW 45485664 Ki = 1.8 nM T32262 C63VLU 45485665 Ki = 7.9 nM T32262 C7VRC1 45485666 Ki = 4.4 nM T32262 CK8Q9R 45485676 Ki = 56 nM T32262 C7SX0U 45485677 Ki = 0.83 nM T32262 C4UB6E 45485687 Ki = 0.26 nM T32262 CQ15ET 45485692 Ki = 0.035 nM T32262 C9LD8A 45487016 Ki = 340 nM T32262 C5AOW0 45487023 Ki = 100 nM T32262 C7HR0U 45487036 Ki = 6.6 nM T32262 CP1W4J 45487037 Ki = 240 nM T32262 C3VJ7P 45487042 Ki = 390 nM T32262 CT5I7G 45487055 Ki = 510 nM T32262 CSL40Y 45487056 Ki = 8900 nM T32262 C5W8NO 45487057 Ki = 41 nM T32262 CQZ4W1 45487059 Ki = 140 nM T32262 CP0A1T 45487060 Ki = 5000 nM T32262 CI9H4P 45487061 Ki = 66 nM T32262 C9AR7C 46174937 Ki = 0.07 nM T32262 C8KSD1 46178835 Ki = 0.3 nM T32262 CK50TO 46232527 Ki = 2511.89 nM T32262 CMFC17 46232562 Ki = 199.53 nM T32262 CCI28M 46232563 Ki = 501.19 nM T32262 C9R2OQ 46232564 Ki = 316.23 nM T32262 CH36RD 46232565 Ki = 1000 nM T32262 CBMT46 46232591 Ki = 158.49 nM T32262 CA0PE5 46232592 Ki = 794.33 nM T32262 C0N4WY 46232593 Ki = 251.19 nM T32262 C7PY3O 46232693 Ki = 199.53 nM T32262 C63ELO 46232777 Ki = 5.012 nM T32262 CPZV08 46232822 Ki = 12.59 nM T32262 C7C6EX 46884946 Ki = 55 nM T32262 C7ZI3U 46884947 Ki = 720 nM T32262 CBD92Q 46884948 Ki = 320 nM T32262 CEKT29 46884999 Ki = 6000 nM T32262 C4QT8V 46885132 Ki = 17 nM T32262 CMIO63 46885133 Ki = 8.9 nM T32262 CW0JG8 46885134 Ki = 1.4 nM T32262 CCHY85 46885135 Ki = 0.3 nM T32262 CX9A1S 46885183 Ki = 0.023 nM T32262 CS52PG 46885184 Ki = 3 nM T32262 CYFJ59 46885185 Ki = 0.41 nM T32262 CDI07R 46885186 Ki = 1.5 nM T32262 CPG38Y 46885242 Ki = 0.55 nM T32262 C8ZGX3 46885243 Ki = 0.52 nM T32262 C6H4GB 46885244 Ki = 0.12 nM T32262 CZJT73 46885245 Ki = 1.3 nM T32262 CPF6D7 46885299 Ki = 0.072 nM T32262 CK63RE 50939479 Ki = 0.046 nM T32262 C5FO7A 50939608 Ki = 0.056 nM T32262 CGSI36 51357585 Ki = 0.081 nM T32262 CJ41BC 51357854 Ki = 4.3 nM T32262 C13CSY 51357855 Ki = 0.67 nM T32262 CC9HW6 51357856 Ki = 0.066 nM T32262 CKPG40 52940673 Ki = 0.037 nM T32262 CTG24I 52940932 Ki = 0.1 nM T32262 CI1CG2 52941862 Ki = 0.11 nM T32262 CJ3AL6 52942173 Ki = 0.12 nM T32262 CY5CR0 52943413 Ki = 0.69 nM T32262 C5QHP1 52944286 Ki = 0.15 nM T32262 CK0Z5Y 52945887 Ki = 12 nM T32262 CBV64H 52947106 Ki = 1.3 nM T32262 C8C5TS 52949562 Ki = 2.2 nM T32262 CHW8L0 54580803 Ki = 0.14 nM T32262 C2FN4O 54580838 Ki = 0.38 nM T32262 C42KGV 54581838 Ki = 2.2 nM T32262 C1OEW2 54581897 Ki = 0.62 nM T32262 C5W4RL 54581909 Ki = 0.14 nM T32262 CW0HC2 54581910 Ki = 0.036 nM T32262 CLI5N2 54582783 Ki = 1 nM T32262 CR3W8B 54582784 Ki = 5.7 nM T32262 CC0WH5 54583774 Ki = 2.5 nM T32262 C4YE3A 54583775 Ki = 2.8 nM T32262 CWQ19D 54583842 Ki = 0.19 nM T32262 CE8XW4 54583843 Ki = 0.05 nM T32262 CWK2I8 54583844 Ki = 0.16 nM T32262 CH9B7I 54584803 Ki = 0.48 nM T32262 C5BF0V 54585731 Ki = 0.04 nM T32262 C0KVY7 54586710 Ki = 0.4 nM T32262 C8QSR1 54586725 Ki = 0.039 nM T32262 CD6XM5 54587752 Ki = 0.61 nM T32262 C8J7YX 54587762 Ki = 0.29 nM T32262 C1IY0P 56944164 Ki = 0.052 nM T32262 C1HYU6 57404496 Ki = 0.071 nM T32262 C1RT4K 57404529 IC50 = 0.064 nM T32262 C5EH8O 57404534 IC50 = 0.2 nM T32262 CC7N4O 57404535 IC50 = 0.019 nM T32262 CGC3T2 57794685 IC50 = 0.77 nM T32262 CXJQ07 57977594 Ki = 0.022 nM T32262 CED2Y9 57977652 Ki = 0.04 nM T32262 C8IWF0 58864250 IC50 = 98 nM T32262 C7F2PL 58864267 IC50 = 100 nM T32262 CDZU21 58864272 IC50 = 700 nM T32262 CY81QW 58864279 IC50 = 1400 nM T32262 CQ4M0I 58864296 IC50 = 36 nM T32262 C6AY0Z 58864297 Ki = 0.048 nM T32262 C05JZT 58864325 IC50 = 80 nM T32262 CZ4QL7 58864368 IC50 = 97 nM T32262 C3DR7Z 58864407 IC50 = 280 nM T32262 C3JQ0W 58864421 IC50 = 73 nM T32262 C41JYE 58864453 IC50 = 130 nM T32262 CN2D3I 58864463 IC50 = 590 nM T32262 C80MGA 58864477 IC50 = 430 nM T32262 CC68UX 58864479 IC50 = 180 nM T32262 CZU98O 58864506 IC50 = 45 nM T32262 C3EM2R 58864520 IC50 = 4500 nM T32262 C3A6HC 58901616 IC50 = 170 nM T32262 CCUA34 59554855 Ki = 64 nM T32262 C1YVE4 59554856 Ki = 0.1 nM T32262 C3EY2M 59554857 Ki = 1880 nM T32262 C0Q8JI 59554867 Ki = 115 nM T32262 C0S5YQ 59554876 Ki = 303 nM T32262 CZ8SB6 59554885 Ki = 40 nM T32262 CK96TS 59554895 Ki = 0.5 nM T32262 C8EAB3 59554924 Ki = 56 nM T32262 CJ87WH 59554934 Ki = 14 nM T32262 CZB69P 59554936 Ki = 18 nM T32262 C75RQS 59554942 Ki = 260 nM T32262 CTKE18 59554947 Ki = 1800 nM T32262 CLY1Q5 59554953 Ki = 54 nM T32262 CKP8E2 59554975 Ki = 8 nM T32262 C36LQX 59554982 Ki = 32 nM T32262 CM7W1X 59554993 Ki = 1 nM T32262 CJF23X 59555008 Ki = 118 nM T32262 C7PKE1 59555012 Ki = 7 nM T32262 CO83KR 59555024 Ki = 68 nM T32262 C3X4RA 59555031 Ki = 0.07 nM T32262 C2S4GJ 59555036 Ki = 3 nM T32262 CVS38C 59555048 Ki = 0.9 nM T32262 C3P8VH 59555055 Ki = 14 nM T32262 CL36VD 59555056 Ki = 124 nM T32262 C0WM7K 59555066 Ki = 1 nM T32262 CJH3B1 59555074 Ki = 2 nM T32262 C9OWC3 59555100 Ki = 20 nM T32262 C57IML 59555102 Ki = 203 nM T32262 CBA7R3 59555111 Ki = 865 nM T32262 CECH35 59555152 Ki = 59 nM T32262 C0O6KE 59555157 Ki = 2 nM T32262 C62BDC 59555187 Ki = 0.02 nM T32262 CD63KR 59555230 Ki = 22 nM T32262 CK8VN2 59555236 Ki = 806 nM T32262 CE1HT0 59555245 Ki = 202 nM T32262 CFI6Z8 59555258 Ki = 10 nM T32262 CO4VJ9 59555260 Ki = 52 nM T32262 C51OYL 59555274 Ki = 763 nM T32262 C42QTA 59555277 Ki = 30 nM T32262 CA9GL6 59555326 Ki = 45 nM T32262 COJ84D 59555331 Ki = 2 nM T32262 CV13OQ 62705051 EC50 = 3 nM T32262 C4YHM2 68857312 EC50 = 0.15 nM T32262 C0GH3B 69747490 Ki = 0.11 nM T32262 CUQ78F 70681261 IC50 = 380 nM T32262 CS0P8G 70681269 IC50 = 220 nM T32262 CD4W6J 70681270 IC50 = 0.12 nM T32262 CA0GP3 70681361 IC50 = 0.1 nM T32262 C83WEP 70681362 IC50 = 0.24 nM T32262 CNA09E 70682193 Ki = 7.2 nM T32262 C9S1RD 70682194 Ki = 250 nM T32262 C78DAT 70683458 IC50 = 3 nM T32262 CPS24M 70683493 IC50 = 0.093 nM T32262 CP09GW 70684297 Ki = 750 nM T32262 CU3F7D 70684299 IC50 = 210 nM T32262 C2GH6T 70685453 IC50 = 32 nM T32262 C4MIR9 70685454 IC50 = 120 nM T32262 CXK7N2 70685565 IC50 = 0.33 nM T32262 CT8CJ5 70685566 IC50 = 0.39 nM T32262 C4F2XL 70685594 IC50 = 6.8 nM T32262 C5Z4TE 70685595 IC50 = 0.28 nM T32262 CUO9N4 70686450 Ki > 1000 nM T32262 C92GRS 70686451 Ki = 1900 nM T32262 CY3F6J 70686453 IC50 = 330 nM T32262 CDZ9Y3 70686454 IC50 = 8500 nM T32262 C4DP6B 70687597 IC50 = 0.049 nM T32262 C06YZS 70687709 IC50 = 4.4 nM T32262 CT6I9A 70687746 IC50 = 6.6 nM T32262 C1VI4M 70688551 Ki > 1000 nM T32262 CL4I8H 70688552 Ki = 2.5 nM T32262 CMJ9P6 70688553 Ki > 1000 nM T32262 COF79Z 70688557 IC50 = 4 nM T32262 CW1U7R 70689654 IC50 = 11 nM T32262 CL2PV7 70689756 IC50 = 0.27 nM T32262 C58NQB 70690613 Ki = 300 nM T32262 C80HOI 70690614 Ki = 1400 nM T32262 C0YA3Z 70690615 Ki = 0.65 nM T32262 CFQ7Z0 70690616 Ki = 16 nM T32262 C4BG7D 70690617 Ki = 250 nM T32262 C8H0NL 70690619 IC50 = 170 nM T32262 C86BMI 70691910 IC50 = 0.33 nM T32262 CND85T 70692757 Ki = 2100 nM T32262 CF1D0A 70692758 Ki > 1000 nM T32262 CRDT90 70692759 Ki = 230 nM T32262 CF4R5I 70692761 IC50 = 860 nM T32262 CKN87D 70693851 IC50 = 99 nM T32262 C5ZC4H 70693987 IC50 = 1.9 nM T32262 COP8L5 70694798 Ki > 1000 nM T32262 CVH1E7 70694802 Ki = 0.55 nM T32262 CV6LI0 70694803 EC50 = 15 nM T32262 C1P7ZJ 70694804 EC50 = 13 nM T32262 C0UPX1 70694861 Ki = 940 nM T32262 CWSV01 70695973 IC50 = 890 nM T32262 CL89KS 70695974 IC50 = 4.6 nM T32262 CP91SM 70696075 IC50 = 0.1 nM T32262 C2LP3E 70696076 IC50 = 12 nM T32262 C5S7CI 70696077 IC50 = 0.24 nM T32262 CSG16Y 70696078 IC50 = 1.2 nM T32262 CDPJ35 70696079 IC50 = 0.042 nM T32262 CBDN32 70696080 IC50 = 1.3 nM T32262 CK42BQ 70696845 Ki = 2400 nM T32262 C62EGB 70696847 Ki = 84 nM T32262 CH4U7X 70696851 IC50 = 1400 nM T32262 CZ4SR9 71569374 Ki = 27 nM T32262 CS2VA3 71569375 Ki = 0.032 nM T32262 C3OM9G 71569532 Ki = 11 nM T32262 C9WNA4 71569533 Ki = 0.015 nM T32262 C6TI0G 72190777 IC50 = 0.39 nM T32262 C85DFY 72190778 IC50 = 0.37 nM T32262 CE8OT0 72191391 IC50 = 0.22 nM T32262 CYO9R8 72191392 IC50 = 0.26 nM T32262 C9VUN4 72191699 IC50 = 2.9 nM T32262 C7Y8BN 73346897 IC50 = 3 nM T32262 CQ58KP 73347057 IC50 = 910 nM T32262 C85OLV 73348402 IC50 = 8 nM T32262 C7JX6P 73348426 IC50 = 14 nM T32262 CS34XQ 73351480 IC50 = 21.9 nM T32262 CJ46SV 73352727 IC50 = 2 nM T32262 C1WD2P 73352946 IC50 = 9 nM T32262 CWS2T8 73352948 Ki = 0.028 nM T32262 CJH08Z 73353203 IC50 = 3548.13 nM T32262 CT7R5K 73355345 IC50 = 1.7 nM T32262 C4G0TL 73356026 IC50 = 11.2 nM T32262 CP7Y1K 73356029 IC50 = 0.5 nM T32262 C0O5XH 73356030 IC50 = 20.2 nM T32262 C6Q2RG 73356952 Ki = 0.017 nM T32262 CHTC49 76310534 Ki = 9 nM T32262 CSUE07 76310551 Ki = 282 nM T32262 C31NWZ 76321477 Ki = 0.03 nM T32262 C7FVX4 76325057 Ki = 297 nM T32262 CSE87P 76332330 Ki = 1 nM T32262 CXB49M 86298538 EC50 = 100 nM T32262 CH2D9L 86298539 IC50 = 25 nM T32262 CTV8B0 118718879 IC50 = 19000 nM T32262 CDLX50 134130160 IC50 = 0.032 nM T32262 CXHY05 135461116 Ki = 26 nM T32262 CHS46O 46905052 Ki = 0.23 nM T32262 D02NMK 44274034 IC50 = 159 nM T32262 D05LMD 16134896 IC50 = 0.5 nM T32262 D05MSG 44593666 Ki = 0.0128 nM T32262 D08GZJ 54580850 Ki = 0.05 nM T32262 D09TDY 23582940 Ki = 0.35 nM T32262 D0B8HD 44274033 IC50 = 29 nM T58674 CB78RO 16130452 Ki = 0.04 nM T58674 C5WNR8 90655646 Ki > 100000 nM T58674 CWS62E 90655648 Ki = 970 nM T58674 C9OBF7 90655650 Ki = 450 nM T58674 C6BAO1 90655652 Ki = 1200 nM T58674 CLU7N6 90655654 Ki = 980 nM T58674 C2ZAV0 90655656 Ki = 180 nM T58674 CZI74U 90655662 Ki = 850 nM T58674 CCZ96Y 90655670 Ki = 1400 nM T58674 C2OQC3 118719137 Ki = 690 nM T58674 C6RSF2 118719138 Ki = 3000 nM T58674 C2FM7S 118719140 Ki = 1500 nM T58674 C9LD4Q 118719142 Ki = 9000 nM T58674 CV5OM7 118719144 Ki = 960 nM T58674 CBSG19 90655672 Ki = 430 nM T29083 D0AF6O 71731823 IC50 = 6 nM T29083 D0OB0F 5328940 IC50 = 358 nM T29083 D0E3TC 44259 IC50 = 1.52 nM T29083 D03BNU 59604787 IC50 > 10000 nM T29083 D0T3ME 156422 IC50 > 30000 nM T29083 CUJR40 10062694 IC50 = 1 nM T29083 CO9KP5 11583459 IC50 > 10000 nM T29083 CU0E8O 11690457 Ki > 2000 nM T29083 CB0AP2 11705863 Ki > 10000 nM T29083 CQG45C 16109001 IC50 = 25000 nM T29083 C1U8XW 16109036 IC50 = 910 nM T29083 CQNP54 24764449 IC50 = 706 nM T29083 CQ3LF1 25226298 IC50 = 494 nM T29083 C3VRO9 44557921 IC50 > 10000 nM T29083 CLS29B 46872626 IC50 > 10000 nM T29083 CEQN27 52936621 Ki > 1000 nM T29083 C8NA4L 53384644 IC50 > 30000 nM T29083 CV63UL 67240318 IC50 > 10000 nM T29083 CPG3A5 86302574 IC50 > 30000 nM T29083 C4X7SD 122192466 IC50 > 10000 nM T29083 C2MD1Q 155513187 IC50 > 10000 nM T29083 D09PTP 57325421 IC50 = 99 nM T29083 D0K5UF 72710568 IC50 = 5 nM T29083 D0R2WK 16038120 IC50 = 569 nM T29083 D0X7IC 53340664 IC50 = 527 nM T59875 D07KSG 2733526 IC50 = 62.2 nM T59875 D0Y2NE 448537 EC50 = 630 nM T59875 CQ0IC4 63062 IC50 = 13 nM T59875 C5GVH1 3035198 IC50 = 13 nM T59875 CQ6I7M 5333661 EC50 = 84 nM T59875 CIQ9M6 5338394 EC50 = 2000 nM T59875 CL0N2I 6864965 EC50 = 2150 nM T59875 CO35ML 6870927 EC50 = 1600 nM T59875 C5DS0Y 6898921 EC50 = 630 nM T59875 C08OAZ 6911476 EC50 = 820 nM T59875 CVH56Y 9649292 EC50 = 7600 nM T59875 CZ86NG 9657428 EC50 = 2300 nM T59875 C1XBH0 11404599 EC50 = 500 nM T59875 C8DS1F 24825443 IC50 = 130 nM T59875 CZ4P8I 24825444 IC50 = 1300 nM T59875 C7PR1H 24825445 IC50 = 200 nM T59875 CZ9O3D 24825446 IC50 = 5 nM T59875 CW43SX 24825447 IC50 = 160 nM T59875 CKW98C 24825448 IC50 = 1000 nM T59875 CN9TA0 24825453 IC50 = 250 nM T59875 CF1H9X 24825454 IC50 = 790 nM T59875 CN9L7G 46916268 IC50 = 2800 nM T59875 C5ZX4B 54597874 IC50 > 10000 nM T59875 C3WUH8 119706729 EC50 = 9100 nM T59875 CV5G4J 134132870 IC50 = 5600 nM T59875 CM3RD1 134133011 IC50 > 10000 nM T59875 C2URL4 134134246 IC50 = 90 nM T59875 CZ8N5V 134134638 IC50 > 10000 nM T59875 C7IH8A 134135221 IC50 = 1300 nM T59875 CHI42Q 134136166 IC50 = 480 nM T59875 CNQU37 134137309 IC50 = 1000 nM T59875 CD7NA5 134138492 IC50 = 77 nM T59875 C7UYJ9 134139141 IC50 > 10000 nM T59875 CO2RS0 134142980 IC50 = 6700 nM T59875 C9YN5F 134143559 IC50 > 10000 nM T59875 CP04WC 134144077 IC50 = 111 nM T59875 C7WJQ2 134144444 IC50 = 1100 nM T59875 CN2UZ9 134144601 IC50 = 5300 nM T59875 CHBD12 134145941 IC50 > 10000 nM T59875 CIR5J4 134146639 IC50 > 10000 nM T59875 CM2G6A 134149343 IC50 = 520 nM T59875 CAJN82 134150366 IC50 = 890 nM T59875 CYG76M 134150509 IC50 = 187 nM T59875 C2CN7S 134152612 IC50 > 10000 nM T59875 C89SMK 134152807 IC50 = 117 nM T59875 C1O0IW 134153257 IC50 = 270 nM T59875 CTLJ74 134153959 IC50 = 3900 nM T59875 C0Z4OD 134155524 IC50 = 79 nM T59875 C58OUX 134155994 IC50 = 20 nM T59875 CW24XE 134156280 IC50 = 1500 nM T59875 C5K8EG 134156559 IC50 = 500 nM T59875 C6M2AG 134156739 IC50 > 10000 nM T59875 CNXJ86 137628681 IC50 = 20 nM T59875 CK1MG4 145963882 EC50 = 2900 nM T59875 CNR74O 145964037 EC50 = 1140 nM T59875 C5ME8W 145964103 EC50 = 300 nM T59875 CA41IJ 145964137 EC50 = 950 nM T59875 CZ8TP7 145964177 EC50 = 5900 nM T59875 CZ2QE5 145964306 EC50 = 1300 nM T59875 CORM23 145964708 EC50 = 1710 nM T59875 CK75QY 145965282 EC50 = 6000 nM T59875 CN76ZF 145965966 EC50 = 6200 nM T59875 CPV40G 145967057 EC50 = 3500 nM T59875 CK5FT2 145970748 EC50 = 4400 nM T59875 C0N3VX 145972148 EC50 = 950 nM T59875 C6HY3P 145973306 EC50 = 3100 nM T59875 C53HNT 145974196 EC50 = 3000 nM T59875 CBO27S 145974510 EC50 = 4300 nM T59875 CNJ9T5 145975180 EC50 = 7000 nM T59875 C03EFZ 145975760 EC50 = 5300 nM T59875 CKTL80 145975927 EC50 = 760 nM T59875 C46ZSN 145976707 EC50 = 8900 nM T59875 C3P9HV 145977071 EC50 = 700 nM T59875 C96MKS 145977115 EC50 = 3200 nM T59875 CDY0S6 145977581 EC50 = 210 nM T59875 C0XYI1 145978085 EC50 = 390 nM T59875 CB4UP0 145978105 EC50 = 6200 nM T59875 CA4WO3 145978362 EC50 = 7900 nM T59875 C25MFD 145978490 EC50 = 810 nM T59875 CZ51WI 155511276 IC50 = 6619 nM T59875 C7VS5G 155511937 IC50 = 40 nM T59875 C9TRH2 155513082 IC50 = 340 nM T59875 CVCK17 155513135 IC50 = 17 nM T59875 C2PU1J 155513315 IC50 = 60 nM T59875 CMQC26 155515404 IC50 = 53 nM T59875 C1S2CU 155516369 IC50 = 421 nM T59875 CP1L3J 155516697 IC50 = 27 nM T59875 C56PVB 155517429 IC50 = 6527 nM T59875 CT72IK 155518795 IC50 = 511 nM T59875 CND3I7 155518873 IC50 = 140 nM T59875 CZW3R9 155519984 IC50 = 5618 nM T59875 CENQ40 155525746 IC50 > 10000 nM T59875 C31VGH 155527588 IC50 = 3017 nM T59875 CSLJ15 155528850 IC50 = 60 nM T59875 C6IAM4 155529788 IC50 = 115 nM T59875 CR0SX8 155533752 IC50 = 354 nM T59875 CYV61X 155534189 IC50 = 3633 nM T59875 C6A4GZ 155534396 IC50 = 2631 nM T59875 C7UL2T 155535280 IC50 = 4333 nM T59875 CC5HJ6 155535796 IC50 = 26 nM T59875 CLNS19 155536017 IC50 > 10000 nM T59875 CB3CY8 155538987 IC50 = 104 nM T59875 C45FZX 155539762 IC50 = 2700 nM T59875 C2CNK3 155540619 IC50 = 1364 nM T59875 CHXK89 155544191 IC50 = 214 nM T59875 C2C5QZ 155547134 IC50 > 10000 nM T59875 CY3N8B 155549927 IC50 > 10000 nM T59875 CA5G2T 155551013 IC50 = 21 nM T59875 C7AJZ5 155559268 IC50 = 50 nM T59875 C9KY5I 155562382 IC50 = 28 nM T59875 CWK95R 155565459 IC50 = 18 nM T59875 CY71WP 155565677 IC50 = 18 nM T59875 CMX67L 155567147 IC50 = 99 nM T59875 D02RQP 6623 IC50 = 4.91 nM T59875 D06JPQ 5497124 EC50 = 130 nM T59875 D09NFD 6852176 IC50 = 79 nM T59875 D0DX8T 5331325 EC50 = 600 nM T81482 CJ6R1L 18445508 IC50 = 199.53 nM T81482 C3HVM7 18445520 IC50 = 31.62 nM T81482 C8OR0L 18445737 IC50 = 3162.28 nM T81482 CM28GF 18445739 IC50 = 63.1 nM T81482 C0TC2X 18445833 IC50 = 630.96 nM T81482 C3VRO9 44557921 IC50 > 10000 nM T81482 CL0OC7 45375855 IC50 = 2511.89 nM T81482 CZXJ98 45483394 IC50 = 125.89 nM T81482 C25NVM 45483417 IC50 = 316.23 nM T81482 C0I2MB 45483418 IC50 = 251.19 nM T81482 C6CJ2N 45483436 IC50 = 794.33 nM T81482 CZOK17 45483447 IC50 = 1000 nM T81482 C1W0AX 45483460 IC50 = 1000 nM T81482 CICD40 45483461 IC50 = 2511.89 nM T81482 CXK2H9 45483468 IC50 = 1584.89 nM T81482 C7MQI8 45483469 IC50 > 10000 nM T81482 CED7U8 45483470 IC50 = 50.12 nM T81482 CBV30W 45483507 IC50 = 501.19 nM T81482 CAL8P6 45483508 IC50 = 794.33 nM T81482 C2UPW3 45483509 IC50 = 1258.93 nM T81482 CA23TC 45483510 IC50 = 7.943 nM T81482 CZC96T 45483513 IC50 = 19.95 nM T81482 C2ABD6 45483530 IC50 = 251.19 nM T81482 C4EZO3 45483716 IC50 = 63.1 nM T81482 CB3N6J 45483717 IC50 = 501.19 nM T81482 CH1S9G 45483725 IC50 = 79.43 nM T81482 CE6K8L 45483734 IC50 > 10000 nM T81482 C4DG0Z 45483735 IC50 > 10000 nM T81482 CXB94H 53466728 IC50 = 17020 nM T81482 CYQ41S 53466951 IC50 = 1863 nM T81482 CX0R1K 53469059 IC50 = 460 nM T81482 CV7C0D 53469060 IC50 = 37 nM T81482 CCKD45 53469061 IC50 = 61 nM T81482 C91STB 53469449 IC50 = 214 nM T81482 CZ1CI3 53469824 IC50 = 12080 nM T81482 CX4H6I 86583042 IC50 > 10000 nM T81482 C4TXF2 118730409 IC50 > 10000 nM T81482 CXC69T 137321158 IC50 = 26 nM T81482 C2MD1Q 155513187 IC50 > 10000 nM T81482 D02LIR 45375987 IC50 = 6.31 nM T81482 D0N4LR 53469448 IC50 = 420 nM T72534 D0E3TC 44259 IC50 = 1.4 nM T72534 D0T3ME 156422 IC50 > 10000 nM T72534 CD3GX5 868252 IC50 = 10310 nM T72534 CIJ62T 874385 IC50 = 2740 nM T72534 C15WJD 1266829 IC50 = 6177 nM T72534 CPG84J 1348122 IC50 = 260 nM T72534 C2HQ4C 5336169 IC50 = 3570 nM T72534 C8PRV6 17149290 IC50 = 3510 nM T72534 C09DHQ 46234348 Ki = 100 nM T72534 CV63UL 67240318 IC50 > 5000 nM T72534 CQL90X 71540618 IC50 = 5 nM T72534 CMZ8G3 71540620 IC50 = 7900 nM T72534 C9QO2P 71540728 IC50 = 26000 nM T72534 CVG8M5 71540729 IC50 = 6300 nM T72534 C03DNB 71540730 IC50 > 1000 nM T72534 CWE32H 71540731 IC50 = 41 nM T72534 C41SPB 71540732 IC50 = 118 nM T72534 CPGE05 71540733 IC50 = 275 nM T72534 C90TFO 71540846 IC50 = 55 nM T72534 CKE1Y8 71540847 IC50 = 63 nM T72534 CV9JK0 71540848 IC50 = 3100 nM T72534 CSJN15 71540849 IC50 = 20 nM T72534 CUWM58 71719137 IC50 = 27000 nM T72534 CPY19I 71720361 IC50 = 5.4 nM T72534 C6HO9M 71720362 IC50 = 290 nM T72534 CZM67T 72703518 IC50 = 158.49 nM T72534 C18QYF 105539853 IC50 = 10 nM T72534 CBZ59D 118701008 IC50 = 15 nM T72534 CLCO61 135398510 IC50 = 2 nM T72534 CWGA76 137530158 IC50 = 39.81 nM T72534 C2E4DP 139592531 IC50 = 125.89 nM T72534 CZ7YS0 146027031 IC50 = 7.943 nM T72534 C2MD1Q 155513187 IC50 > 10000 nM T72534 CE7TI4 155521619 IC50 = 3981.07 nM T72534 CPW4H0 155531070 IC50 = 25118.86 nM T72534 CONB81 155557716 IC50 = 5011.87 nM T72534 D0K0UM 71540619 IC50 = 3 nM T99057 D04XVN 11707110 IC50 = 0.7 nM T99057 D0K8KX 5280343 IC50 > 10000 nM T99057 D0OB0F 5328940 IC50 = 1 nM T99057 D0T5DP 10127622 IC50 = 14 nM T99057 D01CNB 10172827 IC50 = 50 nM T99057 D01IED 11719003 IC50 > 10000 nM T99057 D02UFQ 11620908 IC50 = 1100 nM T99057 D03CHM 44187362 IC50 = 1.81 nM T99057 D07DTV 11338033 IC50 > 10000 nM T99057 D0B9BU 6918454 IC50 = 2 nM T99057 D0E3TC 44259 IC50 = 2.5 nM T99057 D0I3RD 24963252 IC50 = 3.2 nM T99057 D0K0YC 9826528 IC50 = 7 nM T99057 D0M6BD 16719221 IC50 = 160 nM T99057 D0O2FN 16222096 IC50 = 0.9 nM T99057 D0Q4IX 71727581 IC50 > 10000 nM T99057 D0VF6E 1401 IC50 > 50000 nM T99057 D03BNU 59604787 IC50 > 3500 nM T99057 D02GEJ 5326976 IC50 = 10500 nM T99057 C8KED5 4713 IC50 = 2000 nM T99057 C5HUE3 64981 IC50 = 1 nM T99057 C4MNG8 445840 IC50 > 10000 nM T99057 CJ4QI8 885402 IC50 = 200 nM T99057 CQ7PL4 1235170 IC50 > 20000 nM T99057 C4WFP1 1587957 IC50 = 12300 nM T99057 C9EUD2 1839691 IC50 = 8500 nM T99057 C1SVD2 2132479 IC50 = 9000 nM T99057 CKLG52 2726558 IC50 = 410 nM T99057 C2PB6W 2726567 IC50 > 5000 nM T99057 C5GYO1 2730801 IC50 = 300 nM T99057 CAXR02 3338590 IC50 > 5000 nM T99057 CK27AT 3694944 IC50 = 18100 nM T99057 C8IAR2 5281657 IC50 > 100000 nM T99057 CI68PW 5283685 IC50 > 100000 nM T99057 CXK0S6 5283727 IC50 = 48900 nM T99057 C94GRU 5330453 IC50 = 280 nM T99057 C4G9WR 9547398 IC50 > 100000 nM T99057 C76CUP 9547698 IC50 > 100000 nM T99057 CSNH60 9803891 IC50 = 2 nM T99057 CNA9K2 9806897 IC50 = 1.1 nM T99057 CK2J3G 9863776 IC50 = 2.9 nM T99057 CW8V0K 9864418 IC50 > 50000 nM T99057 C18HKQ 9885748 IC50 = 12800 nM T99057 CHF7G5 9890746 IC50 > 30000 nM T99057 C2Y3WG 9907612 IC50 = 4900 nM T99057 C3EUB4 9911005 IC50 > 30000 nM T99057 C07VNB 9930243 IC50 = 6 nM T99057 CJO47T 9948405 IC50 > 10000 nM T99057 CH57ND 9951825 IC50 = 2600 nM T99057 C3I5HT 9978125 IC50 = 6.2 nM T99057 C37GXK 9983303 IC50 = 40 nM T99057 CV8I5X 9999342 IC50 > 10000 nM T99057 CR8DA1 10024683 IC50 > 100000 nM T99057 CLA93G 10047202 IC50 > 100000 nM T99057 C3LCH5 10047545 IC50 > 100000 nM T99057 C2C1BP 10089048 IC50 = 20000 nM T99057 C0Y5PD 10118314 IC50 = 650 nM T99057 CC5Q3G 10135899 IC50 = 7.7 nM T99057 CH4W9D 10139826 IC50 = 2 nM T99057 C3NW6G 10164464 IC50 = 72 nM T99057 CNJ91A 10185285 IC50 = 14 nM T99057 CJ09AO 10185838 IC50 = 29 nM T99057 C5LUV3 10206034 IC50 = 10 nM T99057 CD3OV6 10206158 IC50 = 0.6 nM T99057 C9XBD5 10225656 IC50 = 10 nM T99057 CMN70R 10228676 IC50 = 20 nM T99057 C5TQ7X 10247543 IC50 > 10000 nM T99057 C1AKH9 10303277 IC50 = 8 nM T99057 CN23SU 10324074 IC50 = 7 nM T99057 CK82OA 10345719 IC50 = 25 nM T99057 C4CP7K 10423452 IC50 > 100000 nM T99057 C95LYF 10457505 IC50 > 30000 nM T99057 CHM9I6 10461359 IC50 = 2 nM T99057 C2WQ8M 10473563 IC50 > 10000 nM T99057 CRX6F0 10479082 IC50 = 200 nM T99057 C83QWV 10714343 IC50 > 100000 nM T99057 CJ4P5T 10905857 IC50 > 30000 nM T99057 C3ZE1P 11064594 IC50 = 2500 nM T99057 CV2O1Z 11165133 IC50 = 43 nM T99057 C82QDW 11188772 IC50 = 30 nM T99057 C8G5WP 11210533 IC50 > 30000 nM T99057 C2W5RC 11235063 IC50 > 25000 nM T99057 C0QA8R 11236142 IC50 = 124 nM T99057 C73WRC 11281076 IC50 = 33 nM T99057 CB6OM9 11384425 IC50 = 18 nM T99057 C13CZV 11395411 IC50 = 82 nM T99057 C0HEN9 11418932 IC50 = 6.8 nM T99057 C0APW4 11422034 IC50 > 10000 nM T99057 C58PRM 11439749 IC50 = 14 nM T99057 CDQ31C 11485916 IC50 = 105 nM T99057 CT9V3D 11496376 IC50 = 630 nM T99057 C0QG4W 11523601 IC50 = 118 nM T99057 CRP2U5 11526671 IC50 = 23 nM T99057 C7HMO6 11526786 IC50 > 10000 nM T99057 CO9KP5 11583459 IC50 > 10000 nM T99057 C0WJX2 11603973 IC50 = 2200 nM T99057 C2OMY7 11611241 IC50 = 39 nM T99057 C2HY5O 11613319 EC50 = 49 nM T99057 CGJ2A0 11617424 IC50 = 30 nM T99057 CK34LS 11632737 IC50 > 5000 nM T99057 CWIH62 11633097 IC50 = 9.3 nM T99057 CP4T3N 11669238 IC50 = 45 nM T99057 CJ9KN7 11683817 IC50 > 10000 nM T99057 CZFH19 11689297 IC50 = 15 nM T99057 CSJ69K 11690375 IC50 = 40 nM T99057 CU0E8O 11690457 Ki > 1000 nM T99057 CB0AP2 11705863 Ki > 10000 nM T99057 C9P0VD 11729539 IC50 > 30000 nM T99057 CPN42M 11755998 IC50 = 2.7 nM T99057 CO3QF7 15951576 IC50 = 1200 nM T99057 C7RUN8 15984125 IC50 = 38 nM T99057 C9TU1O 16046126 IC50 > 1000 nM T99057 CZHJ34 16058637 IC50 = 6800 nM T99057 CKV4G1 16079040 IC50 = 1100 nM T99057 CKX2L7 16085320 IC50 = 960 nM T99057 C4V0CW 16126717 IC50 = 28 nM T99057 C5VPH9 16129448 IC50 = 139 nM T99057 C3KB2P 16221892 IC50 = 7.6 nM T99057 CY8B2U 16221995 IC50 = 5.1 nM T99057 C5PXQ4 16222191 IC50 = 6.6 nM T99057 CD3SV4 16222192 IC50 = 5.2 nM T99057 CC5NK6 16222193 IC50 = 16 nM T99057 CX5H2Q 16222302 IC50 = 1708 nM T99057 CR0HT5 16222819 IC50 = 1.8 nM T99057 C6CHI8 16222917 IC50 = 220 nM T99057 CVYD02 16222921 IC50 = 7.2 nM T99057 CF5PJ6 16223027 IC50 = 4.8 nM T99057 C4PVA3 16223325 IC50 = 44 nM T99057 C1AN2Q 16223412 IC50 = 535 nM T99057 C0A5HN 16223413 IC50 = 27 nM T99057 CA80DB 16223418 IC50 = 82 nM T99057 CE2U1Y 16655058 IC50 = 800 nM T99057 C2IF3P 16678352 IC50 = 960 nM T99057 C3IO1C 16679060 IC50 > 10000 nM T99057 CG05KJ 16720763 IC50 = 25 nM T99057 C5FEX0 16727871 IC50 > 5000 nM T99057 CQ79FH 16727872 IC50 > 5000 nM T99057 CP81ZK 16727873 IC50 > 5000 nM T99057 CJ9QN3 16727876 IC50 > 5000 nM T99057 CA6W3J 16727880 IC50 > 5000 nM T99057 C3J4GL 16727881 IC50 = 650 nM T99057 C81MEA 16727889 IC50 = 250 nM T99057 C7UT6L 16727891 IC50 > 5000 nM T99057 CC2XV5 16727892 IC50 > 5000 nM T99057 CN6A7C 16727895 IC50 > 5000 nM T99057 CT0FB2 16727911 IC50 > 5000 nM T99057 C6IM0U 16727912 IC50 > 5000 nM T99057 CO7C9M 16727913 IC50 > 5000 nM T99057 CEF64U 17599247 IC50 = 23100 nM T99057 CAV35B 17903650 IC50 = 26 nM T99057 CNY91P 20791410 IC50 = 33 nM T99057 C1GH5L 20791412 IC50 = 24 nM T99057 CH8A1O 20791416 IC50 = 29 nM T99057 C8KIW5 20791505 IC50 = 48 nM T99057 CZFE08 20791507 IC50 = 76 nM T99057 CKV3A0 20791510 IC50 = 58 nM T99057 C8UTF2 20791535 IC50 = 14 nM T99057 CU36BS 20791561 IC50 > 25000 nM T99057 CP5O8N 20791586 IC50 = 23 nM T99057 C3OTW0 20791598 IC50 = 566 nM T99057 C2WB5M 20791599 IC50 = 331 nM T99057 CKI91V 20791601 IC50 = 203 nM T99057 CV5WM3 20791602 IC50 = 191 nM T99057 C5X3IH 20791605 IC50 = 2650 nM T99057 CR51GI 20791606 IC50 = 5420 nM T99057 CO97JA 20791607 IC50 > 25000 nM T99057 C5EMT7 20791608 IC50 > 25000 nM T99057 CJPS16 20791615 IC50 = 642 nM T99057 CPD4J0 20791616 IC50 = 2320 nM T99057 CB6Z5Q 20791617 IC50 = 1110 nM T99057 CRK28W 20791618 IC50 > 25000 nM T99057 C8BT9L 20791619 IC50 = 68 nM T99057 C15NJF 20791626 IC50 > 25000 nM T99057 CN4W6G 20791639 IC50 = 23 nM T99057 C14YFA 21024387 IC50 = 96 nM T99057 CEQ2L7 21024393 IC50 = 10000 nM T99057 CKPC54 21025113 IC50 = 94 nM T99057 CR8H4Y 21110084 IC50 = 39400 nM T99057 C92GDY 21704772 IC50 = 4.2 nM T99057 CQ7BT0 21704776 IC50 = 33 nM T99057 CZJT36 21704852 IC50 = 5 nM T99057 CO2C7D 21704856 IC50 = 20 nM T99057 CT9N7Z 21808053 IC50 > 5000 nM T99057 CULN54 22025663 IC50 = 19.5 nM T99057 C7X3LY 22179466 IC50 = 147 nM T99057 C69UHM 22179477 IC50 = 36 nM T99057 CJN17H 22179480 IC50 = 6130 nM T99057 C83WSJ 22179488 IC50 = 190 nM T99057 CE35RW 22179532 IC50 = 241 nM T99057 C3CB0X 22179547 IC50 > 25000 nM T99057 CIBU26 22179588 IC50 = 42 nM T99057 CQ2WV5 22179590 IC50 = 14600 nM T99057 C4AKZ1 22179615 IC50 > 25000 nM T99057 CO1D8J 22179618 IC50 = 521 nM T99057 CMKR54 22179638 IC50 = 361 nM T99057 CL9RS7 22179671 IC50 = 181 nM T99057 CI68XT 22179674 IC50 = 18 nM T99057 CY47CN 22179680 IC50 = 168 nM T99057 C2DV7M 22179683 IC50 > 25000 nM T99057 CC6HS9 22179713 IC50 = 397 nM T99057 CXH2L0 22179728 IC50 = 87 nM T99057 COM5D6 22255964 IC50 = 500 nM T99057 CUSD96 22255970 IC50 > 5000 nM T99057 CKO7I9 22255979 IC50 > 5000 nM T99057 C51FVK 22255982 IC50 > 5000 nM T99057 CB13LM 22255988 IC50 > 5000 nM T99057 C8F4NU 22271692 IC50 = 26 nM T99057 CQMO93 22466681 IC50 = 280 nM T99057 CZX61A 22466740 IC50 = 100 nM T99057 C9I8EY 22473189 IC50 = 386 nM T99057 CQRV31 22743091 IC50 = 8 nM T99057 CYUX63 22743123 IC50 = 17 nM T99057 CWQC81 22743127 IC50 = 8 nM T99057 CG6D4M 23647319 IC50 > 10000 nM T99057 CY8Z7X 23647330 IC50 > 10000 nM T99057 C4XD8H 23647348 IC50 > 10000 nM T99057 CN20YH 24743899 EC50 = 6.3 nM T99057 C6JCE7 24753323 IC50 = 28 nM T99057 C50GZI 24753409 IC50 = 53 nM T99057 CC4RZ6 24753410 IC50 = 230 nM T99057 CB3D1Y 24753411 IC50 = 110 nM T99057 C6JF2R 24753412 IC50 = 9 nM T99057 CWX89I 24753603 IC50 = 60 nM T99057 C4CY3V 24753607 IC50 = 110 nM T99057 CFN72M 24753694 IC50 = 64 nM T99057 CQJ2D3 24753784 IC50 = 38 nM T99057 CP1E4R 24753786 IC50 = 99 nM T99057 CA3I4T 24753787 IC50 = 7 nM T99057 CW36DL 24753877 IC50 = 66 nM T99057 COAY09 24753878 IC50 = 97 nM T99057 C9H7EZ 24753971 IC50 = 59 nM T99057 C6CT7I 24753973 IC50 = 26 nM T99057 CS98MR 24754053 IC50 = 46 nM T99057 C9Q3DE 24754054 IC50 = 47 nM T99057 CRJ9G6 24754132 IC50 = 36 nM T99057 CBD59Z 24754133 IC50 = 65 nM T99057 CKV76A 24754134 IC50 = 58 nM T99057 CM8HY9 24754207 IC50 = 4200 nM T99057 C7YG1N 24759534 IC50 = 7200 nM T99057 CM9ED1 24784164 IC50 = 18 nM T99057 C9PA0M 24807809 IC50 > 10000 nM T99057 C61KPI 24856363 IC50 > 50000 nM T99057 C2HEA1 24963248 IC50 = 4.8 nM T99057 CNS0P4 24963250 IC50 = 16 nM T99057 C2Z1GV 24963251 IC50 = 3.2 nM T99057 CF57BL 24963596 IC50 = 8.6 nM T99057 C2F6VC 24965727 IC50 = 26 nM T99057 C9MXU6 24965728 IC50 = 9.8 nM T99057 CQ5K9J 24965731 IC50 = 8.3 nM T99057 CG6PX7 24966075 IC50 = 3.8 nM T99057 CC1AS8 24966426 IC50 = 5 nM T99057 CDJZ34 24966428 IC50 = 4 nM T99057 CNR1E2 24967882 IC50 = 53 nM T99057 CQL29E 24967884 IC50 = 740 nM T99057 CNG6P3 24968231 IC50 = 4.9 nM T99057 CU7W2H 24968572 IC50 = 3.1 nM T99057 CF9UH3 24968575 IC50 = 3.3 nM T99057 C32AUW 25013308 IC50 = 12 nM T99057 C4QF6H 25101222 IC50 = 18000 nM T99057 CVHF49 25124153 IC50 = 17 nM T99057 C7JK8L 25124154 IC50 = 41 nM T99057 C3MUZ7 25124155 IC50 = 14 nM T99057 CI8W7P 25124156 IC50 = 32 nM T99057 CKLW04 25124159 IC50 = 52 nM T99057 C6OSI9 25124477 IC50 = 20 nM T99057 C4A0CP 25124478 IC50 = 76 nM T99057 CPC6N3 25124479 IC50 = 18 nM T99057 CF7BM9 25124819 IC50 = 8.9 nM T99057 CJ56ZC 25125162 IC50 = 54 nM T99057 CD4H7O 25125510 IC50 = 36 nM T99057 CRM79Y 25125842 IC50 = 11 nM T99057 CIUJ83 25167109 EC50 = 45 nM T99057 C6VNB2 25181191 IC50 = 19 nM T99057 CN5TH0 25186684 IC50 = 42 nM T99057 CYHE45 25186685 IC50 = 46 nM T99057 C1B0RC 25186686 IC50 = 20 nM T99057 C6MWK4 25186687 IC50 = 11 nM T99057 CST81A 25186959 IC50 = 32 nM T99057 CM4W6B 25186960 IC50 = 13 nM T99057 CKUI82 25186961 IC50 = 18 nM T99057 C65UMS 25186963 IC50 = 19 nM T99057 CWBI46 25187248 IC50 = 90 nM T99057 CS1F6O 25187538 IC50 = 7 nM T99057 CY07IE 25187543 IC50 = 30 nM T99057 C6DZN3 25187544 IC50 = 13 nM T99057 CZ87LE 25188088 IC50 = 19 nM T99057 C6FGQ1 25206346 IC50 = 1000 nM T99057 CRO09K 25211064 IC50 = 225 nM T99057 C8MBU1 25211459 IC50 = 1800 nM T99057 CF9O0S 25218754 IC50 = 9700 nM T99057 C4T7YX 25218756 IC50 = 13000 nM T99057 CM2GY7 25218822 IC50 = 3 nM T99057 CD80NJ 25218823 IC50 = 4 nM T99057 CT84WC 25218824 IC50 = 8 nM T99057 C6P0UZ 42606202 IC50 = 39 nM T99057 C7NZD9 42606204 IC50 = 25 nM T99057 CWN59K 42606205 IC50 = 94 nM T99057 CCO2Z0 42606316 IC50 = 57 nM T99057 C3ET7Q 42606317 IC50 = 38 nM T99057 CN72OJ 42606318 IC50 = 29 nM T99057 CHG6V0 42606319 IC50 = 109 nM T99057 CQG9O8 42606320 IC50 = 69 nM T99057 CU9E4P 42629114 IC50 > 10000 nM T99057 C48USC 44143344 IC50 = 15000 nM T99057 CM86PK 44143527 IC50 = 750 nM T99057 CC9SL5 44143531 IC50 = 660 nM T99057 CFP1N7 44143534 IC50 = 800 nM T99057 CEL61X 44229839 IC50 = 2100 nM T99057 CYE36B 44241613 IC50 > 40000 nM T99057 C6LG5T 44241614 IC50 > 40000 nM T99057 C90AGP 44279526 IC50 = 1100 nM T99057 C4EI5V 44279624 IC50 = 160 nM T99057 C6M1OS 44279650 IC50 = 3.6 nM T99057 CA0M5Q 44279651 IC50 = 210 nM T99057 CF1X7T 44279777 IC50 > 10000 nM T99057 CWEL07 44279868 IC50 = 550 nM T99057 CF87XG 44279881 IC50 = 3000 nM T99057 CD6CJ8 44279890 IC50 = 110 nM T99057 C5DBE9 44279911 IC50 = 99 nM T99057 C6J1OV 44279943 IC50 = 3300 nM T99057 C7H3PB 44279996 IC50 = 21 nM T99057 CZYS81 44283696 IC50 = 25 nM T99057 CD0EH5 44283728 IC50 = 140 nM T99057 C91FKW 44328166 IC50 = 35 nM T99057 C1PIV3 44328167 IC50 = 450 nM T99057 C68XOD 44328201 IC50 > 10000 nM T99057 CSU37A 44328224 IC50 > 10000 nM T99057 C1HX0W 44328247 IC50 = 68 nM T99057 CKE68U 44328248 IC50 > 10000 nM T99057 CM6B3A 44328249 IC50 = 185 nM T99057 CL5O9W 44328252 IC50 = 680 nM T99057 C65NIO 44328253 IC50 = 125 nM T99057 C0O4XE 44328572 IC50 = 1400 nM T99057 C2IS5Y 44328691 IC50 = 2100 nM T99057 CMW9F0 44328708 IC50 = 1900 nM T99057 CCP8J1 44328755 IC50 = 13500 nM T99057 CO0S3H 44333650 IC50 = 2 nM T99057 CJ16TV 44333771 IC50 = 28 nM T99057 CPC8D0 44333792 IC50 = 212 nM T99057 CH4NW2 44333813 IC50 = 1 nM T99057 C1Y2CA 44333834 IC50 = 2 nM T99057 CZ6OS0 44333854 IC50 = 9 nM T99057 CZ4VX0 44405504 IC50 = 800 nM T99057 CGNY76 44406797 IC50 = 6786 nM T99057 CLG76N 44406798 IC50 = 4496 nM T99057 C74NHO 44407254 IC50 = 3470 nM T99057 C08BQD 44407284 IC50 = 805 nM T99057 C0H6US 44413718 IC50 > 5000 nM T99057 CFYX93 44413976 IC50 = 740 nM T99057 CR6U0N 44413985 IC50 > 2000 nM T99057 CD20CK 44413990 IC50 > 2000 nM T99057 CE9G6B 44413993 IC50 > 5000 nM T99057 CI9AG7 44413998 IC50 = 620 nM T99057 CK6VP8 44414003 IC50 = 1390 nM T99057 CAY1K3 44414006 IC50 = 1440 nM T99057 C5CGN9 44414007 IC50 = 420 nM T99057 CU78XJ 44414009 IC50 = 500 nM T99057 C2O3RA 44414010 IC50 = 500 nM T99057 CCEI57 44414011 IC50 = 430 nM T99057 C8KHP9 44414015 IC50 = 1230 nM T99057 CW1OL5 44414016 IC50 = 350 nM T99057 CY9SE4 44414021 IC50 = 1450 nM T99057 C5Q7KO 44414022 IC50 > 5000 nM T99057 CN02UR 44414024 IC50 = 670 nM T99057 CYK80F 44414025 IC50 > 5000 nM T99057 CB2L1H 44414026 IC50 = 690 nM T99057 CER4G2 44414027 IC50 = 790 nM T99057 CHY41Q 44414028 IC50 = 410 nM T99057 CG60RC 44414372 IC50 = 62 nM T99057 C4TKO7 44414373 IC50 = 73 nM T99057 C7B9EF 44414374 IC50 = 42 nM T99057 CV15GH 44414396 IC50 = 44 nM T99057 CWLQ15 44414397 IC50 = 68 nM T99057 CUL41F 44414398 IC50 = 86 nM T99057 C1YFX2 44414420 IC50 = 220 nM T99057 CT37HL 44414550 IC50 = 510 nM T99057 CPQ83M 44414575 IC50 = 1440 nM T99057 CJAD46 44415333 IC50 > 5000 nM T99057 C06AMS 44415334 IC50 > 5000 nM T99057 C8IL7A 44415335 IC50 > 5000 nM T99057 C1VT7R 44417767 EC50 = 42 nM T99057 CI4JW0 44417768 EC50 = 130 nM T99057 CFN83L 44417769 EC50 = 100 nM T99057 CK73YC 44417770 IC50 = 45 nM T99057 C7TNE3 44417771 IC50 = 150 nM T99057 C6GJD3 44417772 EC50 = 1500 nM T99057 CA05IE 44417773 IC50 = 44 nM T99057 C2IX3Y 44417774 EC50 = 123 nM T99057 C82LKD 44417775 EC50 = 95 nM T99057 CLY7T6 44417776 EC50 = 350 nM T99057 C59VBJ 44417777 EC50 = 30 nM T99057 CN7QO0 44417778 EC50 = 130 nM T99057 CG76RQ 44417779 EC50 = 70 nM T99057 C7TZH3 44417780 EC50 = 88 nM T99057 CLGM87 44417781 EC50 = 330 nM T99057 CJ12MO 44417782 IC50 = 30 nM T99057 C4JG5U 44417783 EC50 = 260 nM T99057 CA8OE1 44417784 IC50 = 26 nM T99057 CAP9Q8 44417785 EC50 = 350 nM T99057 C3OGB8 44417786 EC50 > 10 nM T99057 C51HVW 44417787 EC50 = 100 nM T99057 CFI0Y5 44417788 IC50 = 20 nM T99057 C24RCB 44417789 EC50 > 10 nM T99057 C2YD6G 44417790 IC50 = 145 nM T99057 CZ0C9J 44417791 IC50 = 20 nM T99057 C68HYN 44417792 EC50 = 128 nM T99057 CU3IM9 44417793 IC50 = 85 nM T99057 CSQV34 44417794 EC50 = 37 nM T99057 CPE0C6 44417795 IC50 = 64 nM T99057 CKA7L6 44417796 EC50 = 150 nM T99057 CEJ97B 44417797 IC50 = 37 nM T99057 CV0QD3 44417798 IC50 = 27 nM T99057 CU1NE0 44417799 EC50 = 250 nM T99057 CY5DZ8 44417801 EC50 = 35 nM T99057 CO0L1N 44417802 EC50 = 284 nM T99057 CUK65S 44417804 EC50 = 118 nM T99057 C7PQM6 44417805 IC50 = 298 nM T99057 COBQ43 44417806 EC50 = 43 nM T99057 CAK81N 44417807 IC50 = 46 nM T99057 CE15NX 44417808 EC50 = 54 nM T99057 C8BJ4S 44417809 EC50 = 120 nM T99057 CL81HY 44417810 EC50 = 22 nM T99057 CQU84C 44417812 EC50 = 564 nM T99057 C3HF6D 44417813 EC50 = 694 nM T99057 CP9VZ5 44417814 EC50 = 65 nM T99057 CSH5V7 44417815 EC50 = 6190 nM T99057 C2I7LO 44468504 IC50 = 48 nM T99057 C2VMW6 44469046 IC50 = 182 nM T99057 CKF1D5 44469440 IC50 = 21 nM T99057 CTH3R7 44469586 IC50 = 539 nM T99057 C1TVZ8 44469864 IC50 = 32 nM T99057 C4V6YC 44470284 IC50 = 21 nM T99057 C1SZX9 44545708 EC50 = 0.2 nM T99057 C3VRO9 44557921 IC50 > 10000 nM T99057 CZI8O2 44580056 IC50 = 1500 nM T99057 C4YOF5 44580057 IC50 = 1900 nM T99057 CQL65I 44580058 IC50 = 7600 nM T99057 CV0WF3 44580059 IC50 = 1500 nM T99057 C7Q1VU 44580077 IC50 = 30 nM T99057 CM7DC1 44580107 IC50 = 48000 nM T99057 C5JMS7 44580231 IC50 = 14000 nM T99057 CK1VE7 44580420 IC50 = 400 nM T99057 CEKG17 44580755 IC50 = 21800 nM T99057 CX7E6T 44580756 IC50 = 2400 nM T99057 C5V3PQ 44580757 IC50 = 21200 nM T99057 CXNQ42 44580758 IC50 = 23000 nM T99057 CR9LU0 44580759 IC50 = 49000 nM T99057 C0L9DI 44588712 IC50 = 35 nM T99057 CW2K3V 44588713 IC50 = 36 nM T99057 CM1AR5 44588714 IC50 = 5 nM T99057 CG9CK2 44588732 IC50 = 59 nM T99057 C4IYE2 44588733 IC50 = 55 nM T99057 CNC6I3 44588734 IC50 = 52 nM T99057 CM3Y0O 44588735 IC50 = 26 nM T99057 C3SYC8 44588760 IC50 = 21 nM T99057 CUYD68 44588761 IC50 = 11 nM T99057 CD02AX 44588762 IC50 = 20 nM T99057 CV9ZW5 44588763 IC50 = 10 nM T99057 CZ7LX5 44588812 IC50 = 33 nM T99057 C67ULC 44588813 IC50 = 3 nM T99057 CH13YD 44588814 IC50 = 4 nM T99057 CSTB61 44588815 IC50 = 6 nM T99057 C5Z3LI 44591740 IC50 > 30000 nM T99057 C2DY3A 44603143 EC50 = 0.4 nM T99057 CW2K8V 44603144 EC50 = 3.4 nM T99057 CJ5CH4 44603148 EC50 = 1.3 nM T99057 CO7DT3 44603204 EC50 = 1.5 nM T99057 CMQ0T2 44603207 IC50 = 4546 nM T99057 C4MOE2 44603271 EC50 = 0.6 nM T99057 C87WRB 44603341 EC50 = 0.9 nM T99057 C87FEM 45270051 IC50 > 40000 nM T99057 CU53FK 45273505 IC50 > 40000 nM T99057 CO7Q2F 46186796 IC50 = 15 nM T99057 CBQ3P6 46195697 IC50 = 18 nM T99057 C4U2MA 46196215 IC50 = 36 nM T99057 CUA97D 46209401 IC50 = 3700 nM T99057 C1J6GR 46224908 IC50 > 10000 nM T99057 CZ20AF 49797945 IC50 = 220 nM T99057 C14NZO 49797965 IC50 = 72 nM T99057 C03FHV 49797966 IC50 = 11 nM T99057 CQ4J0V 49797967 IC50 = 20 nM T99057 C4O9ZB 49798006 IC50 = 29 nM T99057 CHSF07 49806372 IC50 > 1000 nM T99057 CB0S2P 49842666 IC50 = 22000 nM T99057 CAI20B 49842778 IC50 = 12000 nM T99057 CRA74I 49842779 IC50 = 17000 nM T99057 CQUS34 51347355 IC50 = 8.7 nM T99057 CEQN27 52936621 Ki > 1000 nM T99057 CM24LF 52938983 IC50 = 18.19 nM T99057 CF04QJ 53318508 IC50 = 5.9 nM T99057 CZY0J7 53323592 IC50 > 100000 nM T99057 C5TED6 53323815 IC50 = 4.6 nM T99057 CNPM14 53341082 IC50 > 3000 nM T99057 C8G4RK 54016394 IC50 = 300000 nM T99057 C9ZFS1 54764923 IC50 > 100000 nM T99057 CT4E8R 56832546 IC50 = 30000 nM T99057 C6O5WH 56951292 IC50 > 10000 nM T99057 CR0Q2N 57523121 IC50 > 10000 nM T99057 C6CUN1 57624898 IC50 = 69 nM T99057 CE23DS 57624909 IC50 = 21 nM T99057 C7F2XZ 57624940 IC50 = 43 nM T99057 CGU9R7 57624954 IC50 = 96 nM T99057 CX8W0C 57624955 IC50 = 14 nM T99057 C6WO3F 57624958 IC50 = 28 nM T99057 C7JFS9 57624960 IC50 = 16 nM T99057 CYA3O4 57625005 IC50 = 63 nM T99057 CW14PM 57625015 IC50 = 99 nM T99057 CGW8C2 57652534 IC50 = 491000 nM T99057 CVK0G4 58056356 IC50 > 50000 nM T99057 CKB3A4 58102283 IC50 = 810 nM T99057 CX1G3L 58102286 IC50 = 210 nM T99057 C6BPR2 58985201 IC50 > 20000 nM T99057 C1R8NM 59139106 IC50 = 29 nM T99057 CB34LP 59139113 IC50 = 56 nM T99057 CWK9I8 59139139 IC50 = 440 nM T99057 CWN47R 59139154 IC50 = 100 nM T99057 CT0JG1 59139161 IC50 = 35 nM T99057 CP5GY6 59139172 IC50 = 190 nM T99057 CL4X3Z 59139185 IC50 = 110 nM T99057 C1PE3R 59139202 IC50 = 2900 nM T99057 CE82OV 59139228 IC50 = 44 nM T99057 C3T5OF 59139235 IC50 = 650 nM T99057 C1J2BP 59139251 IC50 = 27.7 nM T99057 CWO17Q 59139262 IC50 = 11 nM T99057 C5IYT0 59139264 IC50 = 5 nM T99057 CU3PC0 59139312 IC50 = 1190 nM T99057 C91SBH 59139388 IC50 = 940 nM T99057 C62EVK 59139472 IC50 > 50000 nM T99057 CAYO86 59229792 IC50 = 1100 nM T99057 CT3EW2 59292007 IC50 > 1000 nM T99057 CXJ63M 59603829 IC50 = 12000 nM T99057 CQEU96 59603842 IC50 = 120 nM T99057 C1MR8Q 60097495 IC50 > 10000 nM T99057 CMB3A9 66909275 IC50 = 96 nM T99057 C1UVI6 66909316 IC50 = 22 nM T99057 C37NKO 67129970 IC50 > 10000 nM T99057 CK80LJ 67130050 IC50 > 10000 nM T99057 CV63UL 67240318 IC50 > 10000 nM T99057 C7GRV2 68755406 IC50 > 10000 nM T99057 CUC21J 68796122 IC50 = 398.11 nM T99057 C5DGR9 69036886 IC50 = 10000 nM T99057 C51HSA 70791252 IC50 = 37 nM T99057 CEBO91 71452977 IC50 = 980 nM T99057 CUW41T 71460070 IC50 = 801 nM T99057 CB3SO2 71567006 IC50 > 10000 nM T99057 CDJY72 71568837 IC50 = 8600 nM T99057 CRX81Q 71575642 IC50 > 10000 nM T99057 C1AF9L 71579783 IC50 = 63 nM T99057 CGS50U 71579784 IC50 = 13 nM T99057 CIQ0N7 71579876 IC50 = 26 nM T99057 CQW94G 71579877 IC50 = 1000 nM T99057 CXC3S6 71579878 IC50 = 73 nM T99057 CG1QY4 71579965 IC50 = 76 nM T99057 C9CJR7 71579966 IC50 = 54 nM T99057 CZ31PU 71583657 IC50 > 10000 nM T99057 CXSI14 71718330 IC50 > 100000 nM T99057 C1TM3P 71720141 IC50 > 100000 nM T99057 CSVW76 72546488 IC50 = 500 nM T99057 C7HBR1 72546491 IC50 = 5 nM T99057 CXYT34 72546730 IC50 = 29 nM T99057 C1DAW5 72546731 IC50 = 21 nM T99057 C2XZW3 72708899 IC50 > 40000 nM T99057 CKN46T 72708901 IC50 > 40000 nM T99057 C2M8DV 73348939 IC50 = 157000 nM T99057 C6GZ1O 73353368 IC50 = 74 nM T99057 C7M2UX 73356583 IC50 = 25 nM T99057 C3UC9H 73891099 IC50 > 30000 nM T99057 CV8QX0 76310169 IC50 > 30000 nM T99057 CP4ZX2 76317169 IC50 = 240 nM T99057 CA5L4W 76324771 IC50 > 30000 nM T99057 C9GO0P 76328313 IC50 > 100000 nM T99057 C4DT2Z 76335375 IC50 = 85 nM T99057 C39FTZ 76335685 IC50 > 100000 nM T99057 CK61HY 85469442 IC50 = 473 nM T99057 CO2NX0 86294748 IC50 = 1.63 nM T99057 C84NEF 87200366 IC50 = 10 nM T99057 C1HW4B 89735655 IC50 = 1100 nM T99057 C6PHF1 90331409 IC50 > 10000 nM T99057 CW6S8P 90655795 IC50 > 50000 nM T99057 CNYK35 90655796 IC50 = 37000 nM T99057 CE4LR9 90655797 IC50 = 76 nM T99057 CWT2Q8 90656530 IC50 = 56.6 nM T99057 CUYE57 90656531 IC50 = 31.3 nM T99057 CENM20 90656532 IC50 = 142 nM T99057 C2DA8Y 90656533 IC50 = 101.6 nM T99057 CC3VR2 90656534 IC50 = 60.1 nM T99057 C4MN9X 90656535 IC50 = 95 nM T99057 CCJ84Q 90656536 IC50 = 112 nM T99057 C20LEX 90656537 IC50 = 123 nM T99057 CNZ8T1 90656538 IC50 = 138.5 nM T99057 C0DUR3 90656539 IC50 = 314 nM T99057 C9TUH7 90656540 IC50 = 326 nM T99057 C6BQ7R 90656541 IC50 = 411 nM T99057 CW6MU5 90656542 IC50 = 513.2 nM T99057 CW65IY 90656543 IC50 = 559 nM T99057 CUS70J 90656544 IC50 = 773 nM T99057 CU0VP1 90656545 IC50 > 1000 nM T99057 C4CI8E 90656546 IC50 > 1000 nM T99057 C3Q4ER 90656547 IC50 = 5.37 nM T99057 CK5LT8 90656548 IC50 = 11.4 nM T99057 C9JFM0 90656549 IC50 = 44.3 nM T99057 C19KMH 90656550 IC50 = 12.3 nM T99057 C8S2XK 91758407 IC50 > 10000 nM T99057 CG2Y7L 91809196 IC50 > 10000 nM T99057 C0Y8ZK 91933875 IC50 > 1000 nM T99057 C2P3LF 102136592 IC50 = 3400 nM T99057 C6AV2I 117635937 IC50 = 0.5 nM T99057 C4FIN9 117635939 IC50 = 0.019 nM T99057 C1YHR8 118633046 IC50 = 39.2 nM T99057 CLDQ03 118633052 IC50 = 57.5 nM T99057 C5BG4F 118722945 IC50 < 1000 nM T99057 CS1F8W 118722946 IC50 < 1000 nM T99057 C20GTB 118722947 IC50 < 1000 nM T99057 CJ7P1X 118723266 IC50 < 1000 nM T99057 CIH02Q 118723268 IC50 < 1000 nM T99057 C2VO8M 118723269 IC50 < 1000 nM T99057 C6VWT2 118723270 IC50 < 1000 nM T99057 CK63ST 118727694 IC50 = 27.1 nM T99057 CQCX41 118737057 IC50 > 10000 nM T99057 CE6D5X 122181354 IC50 > 1000 nM T99057 C8O7YN 122181355 IC50 > 10000 nM T99057 C8V5HL 122181356 IC50 = 4900 nM T99057 CU4ZK1 122181359 IC50 > 10000 nM T99057 C9LTM2 122181360 IC50 > 10000 nM T99057 CQ94UG 122181362 IC50 > 10000 nM T99057 CAS9U2 122181363 IC50 > 10000 nM T99057 CSON37 122181364 IC50 = 120 nM T99057 CNIA82 122181365 IC50 > 10000 nM T99057 CYDH02 122181366 IC50 = 260 nM T99057 C4X7SD 122192466 IC50 > 10000 nM T99057 CM1JW3 122604219 IC50 > 10000 nM T99057 C2UO3Y 122604256 IC50 > 10000 nM T99057 C65QNK 122604287 IC50 > 10000 nM T99057 CGT97F 122604354 IC50 > 10000 nM T99057 CW0QT8 126480560 IC50 > 10000 nM T99057 CS8C7J 126480561 IC50 > 10000 nM T99057 CCIQ37 126480562 IC50 > 10000 nM T99057 CGY2L4 126480563 IC50 > 10000 nM T99057 CJM59E 126480564 IC50 > 10000 nM T99057 CO9CY8 126480565 IC50 > 10000 nM T99057 CHQ71G 126480566 IC50 > 10000 nM T99057 C2LAM7 126591927 IC50 = 142 nM T99057 CN36JQ 127037910 IC50 = 11 nM T99057 CWL28X 127038287 IC50 = 83 nM T99057 CY95QS 127038614 IC50 = 12 nM T99057 C5S6PX 127038615 IC50 = 15 nM T99057 C04JES 127038616 IC50 = 13 nM T99057 COVZ04 127038617 IC50 = 14 nM T99057 CJ2UY6 127039306 IC50 = 22 nM T99057 CS1N3Z 127039307 IC50 = 28 nM T99057 C8C1DI 127039308 IC50 = 14 nM T99057 CB8TU5 127040913 IC50 = 18 nM T99057 CYG16V 127040980 IC50 = 15 nM T99057 CY9D7F 127040981 IC50 = 94 nM T99057 CJR5F2 127040982 IC50 = 118 nM T99057 CE0CU2 127040983 IC50 = 262 nM T99057 CUZ85G 127041304 IC50 = 345 nM T99057 CD7PL4 127041305 IC50 = 592 nM T99057 C0STZ3 127041603 IC50 = 1900 nM T99057 C58BEO 127041604 IC50 = 127 nM T99057 CUL2T4 127041605 IC50 = 15 nM T99057 CQI1H9 127041606 IC50 = 32 nM T99057 C4KZU9 127041610 IC50 = 941 nM T99057 C4S7BL 127041901 IC50 = 899 nM T99057 CZ6F5V 127042845 IC50 = 81 nM T99057 CM8J6P 127042846 IC50 = 107 nM T99057 C4NFU7 127042847 IC50 = 379 nM T99057 COZA84 127051904 IC50 = 56.7 nM T99057 C3IC2Z 127052212 IC50 = 0.015 nM T99057 C6EXU9 127052827 IC50 = 0.00715 nM T99057 CIU72D 127264586 IC50 = 161 nM T99057 C8ARK0 131801160 IC50 = 142 nM T99057 C0AV5D 131801161 IC50 = 8.5 nM T99057 CL6E4J 132601725 IC50 = 610 nM T99057 CB3C0Z 132819859 IC50 = 16 nM T99057 CK6Z5F 132819860 IC50 = 2500 nM T99057 CR3C9O 132819862 IC50 = 78 nM T99057 CAG60V 132819865 IC50 = 9.8 nM T99057 CE4Z3X 132819866 IC50 = 26 nM T99057 C8IZB3 134129887 IC50 = 4470 nM T99057 C84IXK 134130027 IC50 > 10000 nM T99057 C3TW9Y 134130036 IC50 = 8.2 nM T99057 CTDB31 134130124 IC50 = 6810 nM T99057 CZA37N 134130230 IC50 = 2480 nM T99057 C5N0CA 134130303 IC50 = 9.5 nM T99057 C4S7VK 134130361 IC50 = 1300 nM T99057 C71ATR 134130387 IC50 = 4810 nM T99057 C7U5HA 134130410 IC50 > 10000 nM T99057 C2IB7F 134130412 IC50 = 11 nM T99057 C6BCJ3 134130599 IC50 = 21 nM T99057 CH7A9R 134130612 IC50 = 763 nM T99057 CEH49U 134130924 IC50 = 8.9 nM T99057 COL93E 134131237 IC50 = 1630 nM T99057 C2AN7T 134611886 IC50 > 100000 nM T99057 CXQ03H 135413555 IC50 = 2500 nM T99057 C8GZ2B 135449326 Ki > 4000 nM T99057 C0TE5S 135651612 IC50 = 2200 nM T99057 CYDM01 135891431 IC50 > 10000 nM T99057 CM9NU1 135967827 IC50 = 32 nM T99057 C1FZ5O 135967828 IC50 = 34 nM T99057 CA0F6P 135967829 IC50 = 56 nM T99057 CM5NS2 135988101 IC50 > 2000 nM T99057 C9JH8N 135988105 IC50 > 2000 nM T99057 CZ7EX0 136183413 IC50 = 2450 nM T99057 C01QHB 137348765 IC50 = 1900 nM T99057 C7P4KI 137628642 IC50 = 10.8 nM T99057 CO19HF 137633457 IC50 > 10000 nM T99057 CI1E8V 137634241 IC50 > 10000 nM T99057 CM2VQ1 137636104 IC50 > 10000 nM T99057 CZAM24 137638642 IC50 > 10000 nM T99057 CTI5H6 137641993 IC50 > 10000 nM T99057 CCO7X8 137643676 IC50 > 10000 nM T99057 C07BXP 137644714 IC50 > 10000 nM T99057 CTDK87 137646412 IC50 > 10000 nM T99057 C7D1TY 137647232 IC50 > 10000 nM T99057 CN9A1C 137647463 IC50 > 10000 nM T99057 C5M9VT 137649141 IC50 > 10000 nM T99057 CI46SD 137652179 IC50 > 10000 nM T99057 CC32NU 137654819 IC50 > 10000 nM T99057 C6J5TG 137658266 IC50 > 10000 nM T99057 C4P2JF 137659314 IC50 > 10000 nM T99057 CS61AX 137659496 IC50 > 100000 nM T99057 CK82HJ 141401938 IC50 = 5.7 nM T99057 CKL52O 141401941 IC50 = 7.6 nM T99057 CF3RP1 141401946 IC50 = 3.9 nM T99057 CGQ16R 141401951 IC50 = 29.8 nM T99057 C14JRV 141401954 IC50 > 1000 nM T99057 C3OI7P 141401960 IC50 = 3.4 nM T99057 C89VHZ 141401969 IC50 = 21.5 nM T99057 CW1P4D 141401971 IC50 = 62.8 nM T99057 C1FIE4 145439085 IC50 = 182 nM T99057 CU62AO 145712394 IC50 = 1500 nM T99057 C6VB3O 145925651 IC50 >= 5000 nM T99057 CB06HA 145968373 IC50 > 1000 nM T99057 C73XMU 145968579 IC50 = 6 nM T99057 CQ9TX5 145968636 IC50 = 441 nM T99057 CYQF12 145970111 IC50 > 1000 nM T99057 CFU2Y5 145971060 IC50 = 7 nM T99057 CLT32B 145996530 IC50 = 100 nM T99057 C2MD1Q 155513187 IC50 > 10000 nM T99057 CUXR49 155516714 IC50 = 120 nM T99057 C4NKP6 155518298 IC50 = 1600 nM T99057 C86HPW 155518524 IC50 > 100000 nM T99057 C6EJR2 155526503 IC50 = 158.49 nM T99057 CQCL04 155545442 IC50 = 100 nM T99057 C8SU7Z 155545952 IC50 = 7.7 nM T99057 CCQ36O 155567646 IC50 = 26 nM T99057 D01WAI 135451156 IC50 = 2500 nM T99057 D06KSF 9549300 IC50 > 40000 nM T99057 D08BMM 6312649 IC50 = 2500 nM T99057 D08XVZ 24866313 IC50 > 10000 nM T99057 D0AY0F 70698427 IC50 > 10000 nM T99057 D0DQ6Z 8530 IC50 = 380 nM T99057 D0F0AX 135413546 IC50 = 2500 nM T99057 D0GD8Y 3006531 IC50 = 70 nM T99057 D0I4NN 14056555 IC50 = 2500 nM T99057 D0J3LR 11634725 Ki > 4000 nM T99057 D0M4SY 135440466 IC50 = 182 nM T99057 D0T0VC 2726555 IC50 = 7000 nM T99057 D0TF0V 3085877 IC50 = 2500 nM T99057 D0TY0P 46926364 EC50 = 4 nM T99057 D0V0QJ 389898 IC50 = 380 nM T99057 D0YE1X 9927943 IC50 > 10000 nM T98225 D07XOV 118598754 IC50 = 787 nM T98225 D0E3TC 44259 IC50 = 33.6 nM T98225 D05BVP 3232621 IC50 = 39 nM T98225 D09CDR 77105816 IC50 = 33 nM T98225 D0CC7E 77105818 IC50 = 30 nM T98225 D0JQ0Z 46916176 IC50 = 70 nM T98225 CU80LI 3233012 IC50 = 36 nM T98225 CTM6Q3 3233225 IC50 = 14100 nM T98225 CCBW41 3233247 IC50 = 2200 nM T98225 CHCZ84 3233454 IC50 = 23200 nM T98225 CK48AJ 3233704 IC50 = 31600 nM T98225 C6NMC8 3233824 IC50 = 6540 nM T98225 C3ZBI0 3233960 IC50 = 15800 nM T98225 CW4I6U 3234003 IC50 = 790 nM T98225 C28NYM 3234028 IC50 = 126 nM T98225 CC3UK4 3234462 IC50 = 158 nM T98225 CI63UP 3234644 IC50 = 282 nM T98225 CT8RJ2 3234850 IC50 = 249 nM T98225 C5GE7V 3234998 IC50 = 63 nM T98225 CW4C3P 3235048 IC50 = 7535 nM T98225 COIS18 3235051 IC50 = 22400 nM T98225 C7L9AN 3235086 IC50 = 3550 nM T98225 CU4FQ0 3235202 IC50 = 891 nM T98225 CSJ39A 3235398 IC50 = 891 nM T98225 CGAT36 5327151 IC50 > 1000 nM T98225 CDQ6K1 10943178 IC50 = 29200 nM T98225 CP04JC 11666231 IC50 = 17.8 nM T98225 CR3BS0 12248905 IC50 = 180 nM T98225 CD34SM 12456154 IC50 = 16400 nM T98225 CVYS91 16759572 IC50 = 501 nM T98225 CK0FT2 17757070 IC50 = 178 nM T98225 C4GI3P 44142045 IC50 = 1122 nM T98225 CF4OY0 44142046 IC50 = 631 nM T98225 CT0F8L 44142047 IC50 = 7943 nM T98225 C39AYP 44142048 IC50 > 10000 nM T98225 C18WIG 44142049 IC50 = 3981 nM T98225 CKZ91F 44142050 IC50 = 7943 nM T98225 C37NJT 44142051 IC50 > 10000 nM T98225 CI7K2Y 44142052 IC50 = 126 nM T98225 C9R5PB 44142054 IC50 = 447 nM T98225 CCD0L4 44142055 IC50 = 126 nM T98225 CX65IF 44142058 IC50 = 100 nM T98225 C2EH7D 44142065 IC50 = 1000 nM T98225 CZ5C6G 44142067 IC50 = 178 nM T98225 CI5O6U 44142068 IC50 = 501 nM T98225 CWH16X 44223933 IC50 = 250 nM T98225 CO8N4M 44223937 IC50 = 794 nM T98225 CDF5Y8 44223946 IC50 = 708 nM T98225 CGLQ20 44223952 IC50 = 40 nM T98225 CR6VH2 44223953 IC50 = 35 nM T98225 C2IBW0 44223954 IC50 = 161 nM T98225 CS3Q2Y 44223955 IC50 = 29 nM T98225 C5M1UN 44223957 IC50 = 45 nM T98225 C6E5PK 44223962 IC50 > 10000 nM T98225 CK8G1T 44223965 IC50 = 42 nM T98225 CJ8KD4 44223966 IC50 = 15 nM T98225 CCW0V4 44223967 IC50 = 34 nM T98225 CF78WD 44223968 IC50 = 117 nM T98225 CNE30X 44223970 IC50 = 11 nM T98225 CYR45S 44223971 IC50 = 20 nM T98225 CLZ62P 44223973 IC50 = 12 nM T98225 CIXB09 44223974 IC50 = 47 nM T98225 C2OBX8 44223977 IC50 = 38 nM T98225 C87PSC 44820580 IC50 = 9200 nM T98225 C8O9RB 44820583 IC50 = 13000 nM T98225 C8AE9G 44820584 IC50 = 26000 nM T98225 CT69UN 44820586 IC50 = 23200 nM T98225 C29WFN 44820587 IC50 = 14600 nM T98225 C7TLU8 44820588 IC50 = 29200 nM T98225 C01JUR 44820591 IC50 = 23200 nM T98225 CL8NG3 44820592 IC50 = 41200 nM T98225 CZIF50 44820593 IC50 = 26000 nM T98225 CA9WZ8 44820594 IC50 = 36800 nM T98225 C6DG3M 44820595 IC50 = 16400 nM T98225 CI2J6V 44820597 IC50 = 13000 nM T98225 CM24JB 44820598 IC50 = 29200 nM T98225 CW09EB 44820599 IC50 = 41200 nM T98225 CWFP71 44820600 IC50 = 14600 nM T98225 CWU2K3 44820601 IC50 = 13000 nM T98225 CIWF96 44820602 IC50 = 23200 nM T98225 CEN4F1 44820607 IC50 = 26000 nM T98225 C3JBN1 44968184 IC50 = 29 nM T98225 CYW79D 44968186 IC50 = 14 nM T98225 CAY7V6 44968191 IC50 > 10000 nM T98225 C1RBX2 44968193 IC50 > 10000 nM T98225 C5OYK3 44968199 IC50 = 88 nM T98225 COQ3X5 44968200 IC50 = 331 nM T98225 CBS71N 44968204 IC50 = 3675 nM T98225 C2SI9M 44968206 IC50 = 128 nM T98225 CWY31S 44968208 IC50 = 1642 nM T98225 C2T0EM 44968221 IC50 = 229 nM T98225 C8NA2J 44968224 IC50 = 269 nM T98225 CR8DC5 44968225 IC50 = 120 nM T98225 CV19YK 44968230 IC50 = 81 nM T98225 CD4ZN1 44968231 IC50 = 136 nM T98225 C62LWE 45485136 IC50 = 1000 nM T98225 C83ZHJ 45485144 IC50 = 224 nM T98225 CG81TN 45485152 IC50 = 141 nM T98225 C1R0UV 45485153 IC50 = 111 nM T98225 C76HWN 46172958 IC50 = 13000 nM T98225 C6M9XJ 46172959 IC50 = 23200 nM T98225 CQUI12 46172960 IC50 = 8200 nM T98225 CT03XY 46172961 IC50 = 8200 nM T98225 CB0LE4 46172963 IC50 = 13000 nM T98225 CR74SM 46172965 IC50 = 41200 nM T98225 C16QFN 46172966 IC50 = 3680 nM T98225 C7J0IV 46172968 IC50 = 50 nM T98225 CK7T1I 46172969 IC50 = 4100 nM T98225 CE0W7X 46172970 IC50 = 26000 nM T98225 CB32ET 46172972 IC50 = 5820 nM T98225 CK1TI4 46172975 IC50 = 29200 nM T98225 C2AO9E 46172977 IC50 = 26000 nM T98225 CO90KZ 46172978 IC50 = 10400 nM T98225 CIHP23 46172979 IC50 = 32800 nM T98225 CN26HW 46172980 IC50 = 92 nM T98225 CU5EF1 46172981 IC50 = 9200 nM T98225 CJZ20M 46172982 IC50 = 8200 nM T98225 CLJZ24 46172983 IC50 = 9200 nM T98225 CGH05O 46172984 IC50 = 290 nM T98225 CN58VR 46172985 IC50 = 5200 nM T98225 CA40QS 46172989 IC50 = 29200 nM T98225 C65WIO 46172990 IC50 = 5200 nM T98225 CNJ2X9 46172991 IC50 = 18400 nM T98225 CJ73LE 46172992 IC50 = 9200 nM T98225 CLS29B 46872626 IC50 > 10000 nM T98225 C15EJK 46916169 IC50 = 104 nM T98225 CHG8C4 46916170 IC50 = 50 nM T98225 CI56BA 46916172 IC50 = 37 nM T98225 CSFT47 46916173 IC50 = 241 nM T98225 C93DCO 46916174 IC50 = 199 nM T98225 CZ5DJ4 46916177 IC50 = 79 nM T98225 CXK37B 46916178 IC50 = 141 nM T98225 CL1GW0 46916179 IC50 = 90 nM T98225 CZ6DK4 46916182 IC50 = 257 nM T98225 C8BQ1W 46926509 IC50 = 26020 nM T98225 CR93YO 46926510 IC50 = 2320 nM T98225 C0FN2W 46926512 IC50 = 4630 nM T98225 CCUG10 46926515 IC50 = 86 nM T98225 C9NC6W 46926516 IC50 = 42 nM T98225 CZ1D2A 46926518 IC50 = 20 nM T98225 C7S6HT 46926519 IC50 = 13 nM T98225 CG1K5A 46926520 IC50 = 526 nM T98225 CVF48X 46926521 IC50 = 75 nM T98225 C4ULH5 46926522 IC50 = 9 nM T98225 CPE98Z 46926523 IC50 = 14 nM T98225 C6WLX1 46926524 IC50 = 9284 nM T98225 CIU3B7 46926525 IC50 = 1640 nM T98225 C61LUI 46926526 IC50 = 5450 nM T98225 C0IVD1 46926527 IC50 = 18 nM T98225 CAYI59 49795862 IC50 = 123 nM T98225 C1UQN4 49795863 IC50 = 290 nM T98225 CU8OC0 49795864 IC50 = 290 nM T98225 C7T5HW 49795865 IC50 = 60 nM T98225 C6N8EY 49795866 IC50 = 30 nM T98225 C7XS1Z 49795867 IC50 = 150 nM T98225 CR3LJ9 49795868 IC50 = 40 nM T98225 C5EWG8 49855158 IC50 = 47 nM T98225 CS6N8Z 54581884 IC50 = 1666 nM T98225 CW9AE7 60034150 IC50 = 498 nM T98225 CV63UL 67240318 IC50 > 10000 nM T98225 C21JAS 76853169 IC50 = 270 nM T98225 CU04XY 77105624 IC50 = 71 nM T98225 CTIA65 77105820 IC50 = 690 nM T98225 CKB1P9 77106023 IC50 = 40 nM T98225 CXYW85 77106025 IC50 = 200 nM T98225 C2UDS0 77106026 IC50 = 100 nM T98225 C97SJD 77106027 IC50 = 110 nM T98225 CFQ10R 77106028 IC50 = 57 nM T98225 CO14DP 77106030 IC50 = 22 nM T98225 C9G3PA 77106234 IC50 = 110 nM T98225 CPD27I 77106235 IC50 = 21 nM T98225 CLOR37 77106236 IC50 = 47 nM T98225 C2GLD8 77106237 IC50 = 130 nM T98225 C0GYK1 86765296 IC50 = 220 nM T98225 CS12RU 127031435 IC50 = 31.8 nM T98225 CZD87E 127037084 IC50 = 14 nM T98225 CB9Z0V 127038973 IC50 = 4 nM T98225 C3ORU9 127052113 IC50 = 142 nM T98225 C2LWZ1 129318964 IC50 = 8 nM T98225 C4Z5MQ 131839619 IC50 = 8 nM T98225 CH8DP7 132220479 IC50 = 700 nM T98225 C9C3XT 134163708 IC50 = 125.89 nM T98225 C4QM9O 134397095 IC50 = 102 nM T98225 CQ1K2W 134397387 IC50 = 25 nM T98225 CR08AO 134397388 IC50 = 30 nM T98225 CIN73J 134397390 IC50 = 124 nM T98225 C6I1YX 134397391 IC50 = 648 nM T98225 CQ9D1Z 134397392 IC50 = 31 nM T98225 CUX8N5 134397449 IC50 = 70 nM T98225 CDC39N 134397450 IC50 = 634 nM T98225 C8RN6W 134397451 IC50 = 86 nM T98225 CE1HY2 134397452 IC50 = 28 nM T98225 CIR51J 134397453 IC50 = 50 nM T98225 C72KFM 134397463 IC50 = 77 nM T98225 CT16YX 134397502 IC50 = 61 nM T98225 CI45HZ 134397798 IC50 = 299 nM T98225 CY4D8I 135566504 Ki = 89.6 nM T98225 CG3UZ1 135927974 Ki > 1000 nM T98225 C5J2WV 138728749 IC50 = 99 nM T98225 CVU63L 139582016 IC50 = 610 nM T98225 C8PH9S 139582017 IC50 = 1000 nM T98225 CX05ZN 145979845 IC50 = 147 nM T98225 C2MD1Q 155513187 IC50 > 10000 nM T98225 D00ERW 44444843 Ki > 8951 nM T98225 D06CXU 46926513 IC50 = 4 nM T98225 D0D2FC 2794188 IC50 = 104 nM T98225 D0UI7U 46926514 IC50 = 68 nM T86674 C7KF3V 56964696 IC50 = 7810 nM T86674 CDE10F 56965233 IC50 = 7810 nM T86674 CG6X0V 57394314 IC50 > 250000 nM T63816 D0E3SH 6918837 Ki = 0.6 nM T63816 D0E7PQ 5311 IC50 = 0.047 ug.mL-1 T63816 D0L7LC 5352062 Ki = 20.5 nM T63816 D0Y3KG 3121 IC50 > 2000000 nM T63816 D00FHR 9865515 IC50 > 10000 nM T63816 D01WKZ 53340426 IC50 > 1000 nM T63816 D05KED 53340666 IC50 > 1000 nM T63816 D07FPY 6918877 Ki = 8.5 nM T63816 D09XIZ 11538455 Ki = 0.3 nM T63816 D0B3FV 6445533 IC50 = 1 nM T63816 D0B7CH 4775 IC50 > 2000000 nM T63816 D0E6UZ 54575456 IC50 = 191 nM T63816 D0GE5B 56654642 IC50 > 180000 nM T63816 D0GH3Q 9804992 Ki = 1050 nM T63816 D0L2UQ 49855250 Ki = 16 nM T63816 D0M8FD 4261 IC50 = 510 nM T63816 D0XT6W 6918638 Ki = 15 nM T63816 D0Z4RC 24756910 IC50 = 13.2 nM T63816 D0J8OC 5186 IC50 = 300 nM T63816 D00HXJ 118884610 Ki = 1821 nM T63816 D07KQB 72948227 IC50 = 150 nM T63816 D0CH8Q 56965342 IC50 = 5000 nM T63816 D0L1NO 72722126 IC50 = 10 nM T63816 D0NG9V 72950863 IC50 = 130 nM T63816 D0QX3G 71532921 IC50 > 10000 nM T63816 D0SP7T 72948224 IC50 = 40 nM T63816 D0YN2T 86302836 IC50 = 36 nM T63816 CCK23B 4144 EC50 = 5000 nM T63816 CBIR94 10313 IC50 > 33330 nM T63816 C1N2KZ 88129 IC50 = 170000 nM T63816 CF60JA 220184 IC50 > 33330 nM T63816 C35INR 338818 IC50 = 4160 nM T63816 CH1JD3 419176 IC50 > 2000000 nM T63816 C0Y4WC 614947 Ki > 20000 nM T63816 CU3HS2 1108280 IC50 > 100000 nM T63816 CK8I3T 3432579 IC50 > 33330 nM T63816 CZA83Y 4118131 IC50 > 33330 nM T63816 CV9JS5 4288771 IC50 > 33000 nM T63816 C7KAR5 5353765 EC50 = 1000 nM T63816 CH5FO1 5353767 EC50 = 5000 nM T63816 CT68UM 5353768 EC50 > 25000 nM T63816 CXUP49 5353769 EC50 > 25000 nM T63816 C7RZA4 5353770 EC50 = 1000 nM T63816 C18ENP 6918846 Ki = 8.7 nM T63816 C1RD7E 6918878 IC50 > 10000 nM T63816 CE9LP2 9543539 IC50 > 180000 nM T63816 CJ84NF 9815304 IC50 > 10000 nM T63816 CC0EU7 9828788 IC50 = 25 nM T63816 CH2LR4 9835152 IC50 > 33330 nM T63816 C81EYJ 9923508 IC50 = 4.3 nM T63816 CQG4V8 9924543 IC50 = 1.2 nM T63816 COLN58 9965621 IC50 > 33330 nM T63816 CZL7C8 10017099 IC50 = 100 nM T63816 CL4C9H 10154438 Ki = 2032.6 nM T63816 CU4E9S 10247137 EC50 = 5000 nM T63816 CK3I9Y 10271952 EC50 = 1000 nM T63816 C7RC1E 10309899 IC50 = 4.6 nM T63816 CG9L1R 10435243 IC50 = 642.7 nM T63816 C60QVT 10460379 IC50 = 1181 nM T63816 C9OU5F 10464879 Ki = 806.13 nM T63816 CDY91S 10584105 Ki > 20000 nM T63816 CSMT47 10728039 Ki > 20000 nM T63816 CXEA43 10914552 EC50 = 1000 nM T63816 CK8UV7 11019840 Ki = 10860 nM T63816 C1H9RC 11036226 EC50 = 1000 nM T63816 CHBS32 11068279 EC50 > 25000 nM T63816 CB3N5M 11514394 IC50 > 33330 nM T63816 C24SBP 11657529 IC50 > 10000 nM T63816 CQ32FV 11664499 IC50 = 260 nM T63816 CG9OC4 11682502 IC50 = 207 nM T63816 CYB26W 11688197 IC50 > 1000 nM T63816 CC3GQ0 11700059 IC50 > 10000 nM T63816 C8N9UZ 11724319 EC50 = 10000 nM T63816 CE4Z0Y 11844891 IC50 = 1030 nM T63816 C6JF9E 11844892 IC50 = 1140 nM T63816 CY0WV6 11844893 IC50 = 840 nM T63816 CU0M1E 11947684 IC50 = 510 nM T63816 C9G1BN 11993595 IC50 = 4800 nM T63816 CH5JS7 11993694 IC50 = 220 nM T63816 CR5F6I 12397856 IC50 = 13000 nM T63816 CJ94OC 12542182 Ki = 11641 nM T63816 CXJ5G9 13190582 IC50 > 10000 nM T63816 C06UTF 13507024 IC50 = 2500 nM T63816 C1KR4L 14113324 IC50 = 19000 nM T63816 C15MQN 14113325 IC50 = 16000 nM T63816 C2D1KP 15983982 Ki = 5.3 nM T63816 CA2YF9 15984018 IC50 = 76 nM T63816 CHB82E 15986417 IC50 = 61400 nM T63816 C52EVH 15986418 IC50 = 17100 nM T63816 CS1QO9 15986509 IC50 = 99400 nM T63816 CM3T2E 16049824 IC50 > 1 nM T63816 CFK8J5 16068056 Ki = 7.9 nM T63816 CMQP70 16068495 Ki = 11 nM T63816 CT84XO 16068594 Ki = 6.6 nM T63816 CF3ZG5 16068595 Ki = 6.2 nM T63816 CL60CA 16068912 Ki = 3.6 nM T63816 C9ZQB3 16095102 IC50 > 50000 nM T63816 C80XYC 16095113 IC50 > 50000 nM T63816 CJR3T1 16658996 IC50 > 200000 nM T63816 CFLC70 16659045 IC50 = 540 nM T63816 C5CIB4 16663079 IC50 > 50000 nM T63816 C0ZWD2 17747368 IC50 = 1500 nM T63816 CKM7F9 17747371 IC50 = 30 nM T63816 C5P8QU 18618646 EC50 > 25000 nM T63816 CQHD27 20459443 IC50 = 9130 nM T63816 C3CQ6Z 22986766 EC50 > 25000 nM T63816 CKV50N 22986790 EC50 > 25000 nM T63816 CQ12UX 23626081 IC50 = 56 nM T63816 CLM91R 23634769 IC50 = 33 nM T63816 CS58WE 23634770 IC50 = 1900 nM T63816 CF92AI 23634771 IC50 = 4200 nM T63816 CST70R 23634889 IC50 = 280 nM T63816 CX5N6D 23634890 IC50 = 650 nM T63816 C5F9VA 23634891 IC50 = 970 nM T63816 CE7SO1 23634892 IC50 = 730 nM T63816 C5TH3R 23634893 IC50 = 310 nM T63816 C1WX2K 23634894 IC50 = 220 nM T63816 CN9A3R 23634895 IC50 = 1160 nM T63816 CQ6DC3 23635016 IC50 = 580 nM T63816 CY1PR7 23635017 IC50 = 130 nM T63816 CJYE84 23648185 IC50 = 38 nM T63816 CB8A5Q 23648260 IC50 > 50000 nM T63816 CS9WX8 23649315 IC50 = 220 nM T63816 C4UV3T 24726843 IC50 = 320 nM T63816 C5G7IV 24726844 IC50 = 2500 nM T63816 C8RC9P 24744325 IC50 > 50000 nM T63816 C17GDO 24779722 IC50 = 648 nM T63816 CIO7Q6 24853792 IC50 = 4200 nM T63816 CBN0J5 24853793 IC50 = 6000 nM T63816 CI3B6L 24857909 IC50 = 87 nM T63816 CQC8T7 24882475 IC50 = 20 nM T63816 CS1MH8 24888322 IC50 = 18000 nM T63816 C5B0IJ 25023793 IC50 = 33 nM T63816 CHE82I 25023795 IC50 = 1700 nM T63816 CX8G3W 25023796 IC50 = 180 nM T63816 CVRS37 25023797 IC50 = 510 nM T63816 C7GO3U 25023798 IC50 = 170 nM T63816 C3G2AU 25023799 IC50 = 70 nM T63816 CAS18V 25023800 IC50 = 350 nM T63816 CX7D5B 25023801 IC50 = 130 nM T63816 CZG50I 25023802 IC50 = 320 nM T63816 CF9WH6 25023808 IC50 = 420 nM T63816 CVS1M4 25023811 IC50 = 970 nM T63816 C2O9CE 25023812 IC50 = 3500 nM T63816 CW6KR2 25023813 IC50 = 2700 nM T63816 C10CNP 25023814 IC50 = 9400 nM T63816 C5IJ6X 25023815 IC50 = 340 nM T63816 C24MTU 25023816 IC50 = 2500 nM T63816 CKY94C 25023817 IC50 = 3300 nM T63816 CJG8C5 25023818 IC50 = 760 nM T63816 CLA50V 25023819 IC50 = 850 nM T63816 CV8EF6 25032862 IC50 > 50000 nM T63816 CX69SY 25066355 IC50 = 2580 nM T63816 CF8VP4 25066356 IC50 = 1200 nM T63816 CS9XH7 25066547 IC50 = 1250 nM T63816 C46AGN 25066548 IC50 = 159 nM T63816 CJF2M7 25066549 IC50 = 447 nM T63816 CT08NK 25141401 IC50 = 1100 nM T63816 CB4E2J 25155956 IC50 > 50000 nM T63816 CFS5O4 25168576 IC50 = 75 nM T63816 C0R5OK 25168856 IC50 = 30 nM T63816 CCD5M7 25227504 IC50 = 79.4 nM T63816 CK0D5S 25227505 IC50 = 284 nM T63816 CN97JP 25227508 IC50 = 118 nM T63816 CW8R1B 25227513 IC50 = 454 nM T63816 C43BHY 25269097 IC50 = 319 nM T63816 C2LES7 42599455 IC50 = 3.7 nM T63816 C2KO0F 42599456 IC50 = 5.3 nM T63816 C1UAO7 42601485 IC50 > 50000 nM T63816 CDT65Y 42631047 IC50 > 100000 nM T63816 CO57GS 44138033 IC50 = 12900 nM T63816 CAG5L0 44228659 IC50 = 550 nM T63816 CY0QB9 44253226 IC50 = 127 nM T63816 CL80GX 44328682 EC50 > 25000 nM T63816 CWY06M 44363182 IC50 = 2.7 nM T63816 CN91KP 44363187 IC50 = 0.3 nM T63816 C3U8EF 44442437 IC50 = 180 nM T63816 C9ZUW5 44442438 IC50 = 98 nM T63816 CJ6SN4 44442439 IC50 = 2100 nM T63816 CP71RI 44445956 IC50 = 24 nM T63816 C3KLP5 44445957 IC50 = 23 nM T63816 CF9RX6 44445958 IC50 = 33 nM T63816 CNC51G 44447194 IC50 > 50000 nM T63816 C8WKU9 44453790 IC50 = 4 nM T63816 C5VP4D 44454144 IC50 > 50000 nM T63816 C4FKU6 44541235 IC50 = 35 nM T63816 C7F8YJ 44543715 Ki = 17500 nM T63816 CW4KH2 44551271 IC50 = 3000 nM T63816 C17BGM 44561972 IC50 = 4890 nM T63816 C04SOM 44561973 IC50 = 12910 nM T63816 C5RD6F 44561974 IC50 = 6030 nM T63816 CA7CG3 44561975 IC50 = 4040 nM T63816 C3UV7C 44561976 IC50 = 4380 nM T63816 C61AMY 44562034 IC50 = 4310 nM T63816 C4HQ8S 44562035 IC50 = 8190 nM T63816 C7PKX5 44562036 IC50 = 7680 nM T63816 C92FSV 44562037 IC50 = 22780 nM T63816 CX6NB4 44562038 IC50 = 47170 nM T63816 CV28HM 44562039 IC50 = 57060 nM T63816 C5CTG9 44562040 IC50 = 74240 nM T63816 CT65QO 44562076 IC50 = 85600 nM T63816 C3P0TE 44562077 IC50 = 49280 nM T63816 CCUP97 44562078 IC50 = 42810 nM T63816 CG3P8O 44562079 IC50 = 50580 nM T63816 CU92TP 44562080 IC50 = 10250 nM T63816 CW42BX 44562604 IC50 = 110 nM T63816 CDW54Z 44562605 IC50 = 270 nM T63816 C1WY8L 44562606 IC50 = 95 nM T63816 C9MB4K 44562607 IC50 = 450 nM T63816 CH2NP3 44562608 IC50 = 280 nM T63816 CBYZ26 44562609 IC50 = 320 nM T63816 CZU3I7 44562657 IC50 = 200 nM T63816 C3QSI4 44562762 IC50 = 220 nM T63816 CRJS52 44562763 IC50 = 120 nM T63816 C2LH1N 44562764 IC50 = 240 nM T63816 CJ5US8 44562765 IC50 > 2000 nM T63816 CUT7L8 44562766 IC50 = 90 nM T63816 CH2KM0 44562767 IC50 = 70 nM T63816 CQX1R2 44562798 IC50 = 590 nM T63816 CQ5RJ3 44562799 IC50 = 15 nM T63816 C96LVR 44562800 IC50 = 60 nM T63816 CDY0E1 44562801 IC50 = 15 nM T63816 CEM91G 44562802 IC50 = 260 nM T63816 CEA9D0 44562840 IC50 = 60 nM T63816 C3DMN0 44563197 IC50 = 243 nM T63816 CGF8R5 44563236 IC50 = 110 nM T63816 CT63QG 44563237 IC50 = 420 nM T63816 CIO34V 44564642 Ki = 10 nM T63816 CA6Q9Y 44592060 IC50 = 11900 nM T63816 C5H8RA 44598536 IC50 > 10000 nM T63816 CC2QV9 44623002 IC50 > 50000 nM T63816 CVJ51M 44623152 IC50 > 50000 nM T63816 C6TJ2G 44623153 IC50 > 50000 nM T63816 CO7S9W 44626297 IC50 = 210 nM T63816 CE47ZB 45102716 IC50 > 50000 nM T63816 CJWF93 45102721 IC50 > 50000 nM T63816 CSM1O6 45271073 IC50 = 150000 nM T63816 C96ROY 45482635 IC50 > 10000 nM T63816 CV74KP 45482658 IC50 > 10000 nM T63816 CHC0Y1 45482667 IC50 = 1910 nM T63816 CD57RJ 46197798 IC50 = 28 nM T63816 CR04HA 46197799 IC50 = 38 nM T63816 C7V1RE 46216758 IC50 = 5.4 nM T63816 CZ0F6R 46216759 IC50 = 5.5 nM T63816 C0RQ1B 46216760 IC50 = 4.5 nM T63816 CI06QG 46216772 IC50 = 5 nM T63816 C5U7GY 46230638 IC50 = 12 nM T63816 CG2R9Z 46838751 IC50 = 4900 nM T63816 C4B7YX 46838752 IC50 = 3000 nM T63816 C69UBY 46861822 IC50 = 9600 nM T63816 C8D4XL 46861823 IC50 = 10650 nM T63816 CPSI47 46890583 Ki = 6 nM T63816 C90NYX 46896338 IC50 = 13000 nM T63816 CI8ZX5 49799582 IC50 = 7500 nM T63816 CL7PS1 49831258 IC50 > 50000 nM T63816 CI5L2P 49846123 IC50 = 14624.7 nM T63816 C4DL0M 49847150 IC50 = 5730 nM T63816 CC7Y9U 49850262 IC50 = 1100 nM T63816 C50PXU 49855444 IC50 > 50000 nM T63816 C78GKN 53361474 IC50 = 379 nM T63816 CNB63X 53361475 IC50 = 432 nM T63816 CQ43VH 53363518 Ki = 2.4 nM T63816 C6Y2EV 53374826 IC50 > 100000 nM T63816 CYQV72 54030066 IC50 = 310 nM T63816 C0ZK7I 54576529 IC50 > 10000 nM T63816 CTP2S1 54576530 IC50 > 10000 nM T63816 CS8HY5 54576744 IC50 > 10000 nM T63816 C5A7MU 54613496 IC50 = 279 nM T63816 CQ1EX7 54770442 IC50 > 10000 nM T63816 C7OJ4K 56602459 IC50 = 37220 nM T63816 CSY2L7 56602461 IC50 = 42000 nM T63816 CIO96M 56659403 IC50 > 100000 nM T63816 CT4ZY0 56661203 IC50 = 5 nM T63816 C8XKD9 56664649 IC50 = 152 nM T63816 CL18NI 56666337 IC50 > 100000 nM T63816 C9LC5Y 56673234 IC50 > 100000 nM T63816 CWH5N4 56673261 IC50 > 100000 nM T63816 C0ZJG3 56676500 IC50 = 22000 nM T63816 CFUT54 56682413 IC50 = 18000 nM T63816 CZ25SN 56935695 IC50 > 30000 nM T63816 C41ZBJ 56951446 Ki > 50000 nM T63816 C1R7HZ 56951447 Ki > 50000 nM T63816 CP4EL2 57328394 IC50 = 10000 nM T63816 C60XUA 57336554 Ki > 50000 nM T63816 C58USD 57336555 Ki > 50000 nM T63816 C4DZ0B 57336556 Ki > 50000 nM T63816 C7JCL9 57336558 Ki > 50000 nM T63816 CN9W2G 57336559 Ki > 50000 nM T63816 C10DMC 57336560 Ki > 50000 nM T63816 CLR1C6 57336561 Ki > 50000 nM T63816 CU6B5H 57336562 Ki > 50000 nM T63816 CWTK67 57336564 Ki > 50000 nM T63816 C95REB 57336565 Ki > 50000 nM T63816 CU68CZ 57336566 Ki > 50000 nM T63816 C0JQ2U 57336567 Ki > 50000 nM T63816 C8O0CH 57336568 Ki > 50000 nM T63816 C5CN3K 57336569 Ki > 50000 nM T63816 CO0RD1 57336570 Ki > 50000 nM T63816 CDK61Y 57336571 Ki > 50000 nM T63816 C0BT1I 57336572 Ki > 50000 nM T63816 C8ZBR3 57401090 Ki > 50000 nM T63816 C4LI0D 57521296 IC50 = 20 nM T63816 CA5Q6O 58147189 IC50 > 50000 nM T63816 C4DYC0 58147224 IC50 > 50000 nM T63816 CMP04X 58147302 IC50 > 50000 nM T63816 CLD40J 58465708 IC50 > 50000 nM T63816 C1MB4Q 59323957 IC50 > 30000 nM T63816 CK6LX0 59454220 IC50 = 46000 nM T63816 C2SDN1 59454252 IC50 = 36000 nM T63816 CO6A2S 59585196 IC50 = 71000 nM T63816 CP2SF9 60148645 IC50 = 48000 nM T63816 CPZ5Q3 60148646 IC50 = 2600 nM T63816 CPIN79 60148647 IC50 = 1800 nM T63816 CV54QY 60148648 IC50 = 30 nM T63816 C67VHS 60148666 IC50 = 1100 nM T63816 CP2HK9 60148667 IC50 = 20 nM T63816 CXIG57 60148671 IC50 = 340 nM T63816 CKG35S 60148672 IC50 = 300 nM T63816 C8ZL3J 60148690 IC50 = 280 nM T63816 C4KR0W 60148692 IC50 = 390 nM T63816 CK5N4E 60148693 IC50 = 20 nM T63816 C6L4RH 60148695 IC50 = 300 nM T63816 C27DKW 60148711 IC50 = 50 nM T63816 CS2E6C 60148712 IC50 = 100 nM T63816 C2M8ZY 60148714 IC50 = 80 nM T63816 C7JF5U 60148716 IC50 = 80 nM T63816 CCOG03 60148735 IC50 = 60 nM T63816 C8M5GS 60148736 IC50 = 100 nM T63816 C1GX5E 60148737 IC50 = 140 nM T63816 CI9Z3H 60148738 IC50 = 510 nM T63816 C50AXJ 60148739 IC50 = 460 nM T63816 CL5RU7 60148765 IC50 = 1800 nM T63816 C4TQ2N 60148766 IC50 = 330 nM T63816 C5OGC0 60148783 IC50 = 150 nM T63816 CNK4Z9 60148788 IC50 = 50 nM T63816 C4SJ0G 60148789 IC50 = 290 nM T63816 C35CSJ 60148809 IC50 = 230 nM T63816 CNL3D0 60148834 IC50 = 500 nM T63816 CXV45D 60148836 IC50 = 4400 nM T63816 C6NF5L 60148861 IC50 = 100 nM T63816 CCB9L4 60148862 IC50 = 40 nM T63816 CA8YU9 60148950 IC50 = 60 nM T63816 CPF50R 60148997 IC50 = 340 nM T63816 CB7X2E 60151224 IC50 > 10000 nM T63816 CY05OU 60151225 IC50 > 10000 nM T63816 CWO8H0 60152596 IC50 > 10000 nM T63816 CQ1U0P 60200243 IC50 = 5900 nM T63816 CBN3L0 69950064 Ki = 75 nM T63816 C6RFQ8 70676597 IC50 > 20000 nM T63816 CE67KO 70695508 IC50 = 110000 nM T63816 CQY1I6 70789579 Ki = 23800 nM T63816 C0ES2V 71453199 IC50 = 1200 nM T63816 C6C4OT 71458560 IC50 = 5.9 nM T63816 C0KRN9 71458561 IC50 = 3 nM T63816 C2HZ7Q 71460412 IC50 = 99 nM T63816 CBK53U 71462097 IC50 = 120 nM T63816 C1MH5Z 71467962 IC50 = 184.67 nM T63816 CJU64Z 71468161 IC50 = 157.79 nM T63816 C0CX7P 71476624 Ki = 6115 nM T63816 C6QPH1 71476625 Ki = 990.23 nM T63816 C3JLD4 71476626 Ki = 8361 nM T63816 C3OH6T 71476627 Ki = 11204 nM T63816 CFQ2N9 71520536 IC50 > 10000 nM T63816 C0LWJ6 71520631 IC50 = 16.3 nM T63816 CO28HI 71520716 IC50 = 82.6 nM T63816 CVA5Q7 71520717 IC50 = 11.9 nM T63816 C89SWX 71527724 IC50 > 30000 nM T63816 CDW81Y 71574856 IC50 > 33330 nM T63816 CX01BJ 71574948 IC50 > 33330 nM T63816 CO8YU7 71574949 IC50 > 33330 nM T63816 CX6I3N 71577043 IC50 = 140 nM T63816 CKR6U8 71583101 IC50 = 1500 nM T63816 CBZ5S9 71583103 IC50 = 1600 nM T63816 C3PSJ9 71583105 IC50 = 1900 nM T63816 C7HG0K 71655802 IC50 = 21800 nM T63816 CPJ4V7 71680913 IC50 > 33000 nM T63816 C9X8KM 71680914 IC50 > 33000 nM T63816 C4W2MA 71680915 IC50 > 33000 nM T63816 C3KO9V 71680916 IC50 > 33000 nM T63816 CN4X5O 71680917 IC50 > 33000 nM T63816 CWAM13 71680918 IC50 > 33000 nM T63816 CI9G3B 71681069 IC50 = 14000 nM T63816 CIR56T 71721558 IC50 > 100000 nM T63816 CCD18W 71721946 IC50 > 100000 nM T63816 CFUC24 71722010 IC50 > 10000 nM T63816 C6U9VB 71769925 IC50 = 10730 nM T63816 CIRH21 71769926 IC50 = 10630 nM T63816 C26HDR 71769927 IC50 = 3960 nM T63816 C5RXY7 71769928 IC50 = 7260 nM T63816 CT1RZ2 71770054 IC50 = 12320 nM T63816 CTPJ18 71770057 IC50 = 11250 nM T63816 C1TSQ4 71770058 IC50 = 50560 nM T63816 CVU1W6 71770059 IC50 = 68110 nM T63816 CHK58Q 71770060 IC50 = 12290 nM T63816 CG3X4E 71770191 IC50 = 13220 nM T63816 CJ87KH 71770193 IC50 = 12640 nM T63816 C8J7IV 71770194 IC50 = 5721 nM T63816 CN5D6Z 71770321 IC50 = 9070 nM T63816 C13MPI 71770439 IC50 = 19950 nM T63816 C5K4ZC 71770562 IC50 = 52450 nM T63816 CT7L6G 72163687 Ki > 20000 nM T63816 CKE9D3 72163688 Ki > 20000 nM T63816 CI9H6L 72164895 IC50 = 3982 nM T63816 CS5UL7 72195322 IC50 = 81500 nM T63816 CV09DJ 72734543 IC50 > 1000 nM T63816 CJ4IN2 72948223 IC50 = 120 nM T63816 CEV08B 72948226 IC50 = 110 nM T63816 COCR40 72948414 IC50 = 230 nM T63816 CX3W1T 73333311 IC50 = 15000 nM T63816 C21XQI 73345596 IC50 = 190 nM T63816 C5FDJ0 73347611 IC50 = 28 nM T63816 CSP58Q 73353181 IC50 = 610 nM T63816 CGM2S4 73356727 IC50 = 18 nM T63816 CZB6G7 73776472 IC50 = 5700.7 nM T63816 C2KUJ9 76310312 IC50 = 20 nM T63816 C7ZM6V 76310313 IC50 = 330 nM T63816 C31XNE 76310314 IC50 = 670 nM T63816 CLM96R 76313986 IC50 = 150 nM T63816 CBCU49 76313987 IC50 = 80 nM T63816 CKW35L 76317533 IC50 = 410 nM T63816 COC82G 76317534 IC50 > 50000 nM T63816 CKC9E0 76321252 IC50 = 7100 nM T63816 CGZ47O 76321253 IC50 = 200 nM T63816 C2ODF9 76321254 IC50 = 530 nM T63816 CP52FW 76324875 IC50 = 30 nM T63816 CTRP59 76324876 IC50 = 40 nM T63816 C89AOG 76324877 IC50 = 60 nM T63816 CM6H9C 76324878 IC50 = 20 nM T63816 C6VG7C 76332116 IC50 > 50000 nM T63816 CH9DC2 76332117 IC50 = 904000 nM T63816 CTZ53J 76332759 IC50 = 38040 nM T63816 CKI74A 76853213 IC50 > 20000 nM T63816 C0ZKI5 76853285 IC50 = 14 nM T63816 CCR7L2 76853289 IC50 > 100000 nM T63816 CJ6Z0X 78324068 IC50 > 20000 nM T63816 C3U0KE 81689842 IC50 = 54 nM T63816 CG5ZD9 86291495 IC50 = 58 nM T63816 C61VCD 86294741 IC50 = 100000 nM T63816 CBWV30 86294747 IC50 = 64000 nM T63816 C06YBD 86302594 IC50 = 75900 nM T63816 C3EM7H 86581004 IC50 = 120 nM T63816 C7UK3Y 86581005 IC50 = 63 nM T63816 CY64UM 86581152 IC50 = 120 nM T63816 CY5V7C 86581153 IC50 = 47 nM T63816 C1HE8I 86581432 IC50 = 2000 nM T63816 CZM07I 86581434 IC50 = 380 nM T63816 C8ZQG9 86581435 IC50 = 220 nM T63816 CS5I4Y 87261507 IC50 = 1080 nM T63816 CYW51P 90654946 IC50 = 40100 nM T63816 CJH1S6 90654947 IC50 > 100000 nM T63816 CSR56C 90655296 IC50 = 71500 nM T63816 CSDO81 90664458 Ki = 16 nM T63816 CI9M0E 90665809 IC50 = 46970 nM T63816 C23GNF 90665810 IC50 = 58880 nM T63816 CY0P7X 90665811 IC50 = 132500 nM T63816 CJO6T1 91810840 IC50 = 2200 nM T63816 C0FCU9 91938063 IC50 = 31.54 nM T63816 C34WIG 92045024 IC50 > 100000 nM T63816 C9OC0F 101882265 IC50 = 67800 nM T63816 C7PS2E 102140473 IC50 = 9.3 nM T63816 C3PFY8 102140474 IC50 = 37 nM T63816 C12GJX 102366363 IC50 > 20000 nM T63816 CO25LD 102366364 IC50 = 7800 nM T63816 C8CER4 102366365 IC50 > 20000 nM T63816 CT7Z8F 102514716 IC50 = 19730 nM T63816 CS2UL0 117829456 IC50 = 78 nM T63816 C7L4OT 117829461 IC50 = 280 nM T63816 C50VUN 117829462 IC50 = 86 nM T63816 CSU52M 118656852 IC50 = 1200 nM T63816 CB6AJ9 118656853 IC50 = 600 nM T63816 C3KAM7 118681924 IC50 = 17 nM T63816 CK6YX4 118706143 IC50 = 41 nM T63816 C8JMF2 118706144 IC50 = 26 nM T63816 CZY1Q2 118706145 IC50 = 31 nM T63816 CC3LG6 118706146 IC50 = 15 nM T63816 CVCM47 118706554 IC50 = 10.3 nM T63816 C98SPM 118706555 IC50 = 8.3 nM T63816 CB8Q2L 118706556 IC50 = 4.2 nM T63816 CV3ST1 118706557 IC50 = 11 nM T63816 CAF41G 118707835 IC50 > 20000 nM T63816 C0P4EV 118707836 IC50 = 15200 nM T63816 CC8KL3 118707837 IC50 > 20000 nM T63816 C9VI8U 118707838 IC50 > 20000 nM T63816 CRU9G3 118707839 IC50 > 20000 nM T63816 C9SWI4 118707840 IC50 > 20000 nM T63816 CW9UJ1 118707841 IC50 > 20000 nM T63816 CBYI69 118707842 IC50 > 20000 nM T63816 CXF0U3 118714375 IC50 = 86400 nM T63816 C2M5OR 118714376 IC50 = 56300 nM T63816 CY4GN9 118714377 IC50 = 83100 nM T63816 CRL92Y 118714414 IC50 = 9800 nM T63816 CR37MV 118714415 IC50 = 7600 nM T63816 CUI51W 118720529 IC50 = 440.3 nM T63816 C1EC5S 118721286 IC50 = 43 nM T63816 CI8G4X 118737400 IC50 = 11700 nM T63816 C2F8TQ 118737455 IC50 = 30 nM T63816 CZ61KV 118753026 IC50 = 230 nM T63816 CFI23Y 118753027 IC50 = 1000 nM T63816 C75LTK 118753189 IC50 = 4600 nM T63816 C5L8QM 118884518 IC50 = 20500 nM T63816 CB84TO 121278998 IC50 = 1900 nM T63816 C9S5OK 121279020 IC50 > 50000 nM T63816 CL3M2F 121499152 IC50 > 33330 nM T63816 C28JVO 122192004 IC50 > 10000 nM T63816 CF2D8U 122192005 IC50 > 10000 nM T63816 C3V5ND 122550211 IC50 > 10000 nM T63816 CZE35C 122648343 IC50 > 1000 nM T63816 C54RNT 122648367 IC50 > 1000 nM T63816 C1UVI7 122648600 IC50 > 1000 nM T63816 CMX59K 122648648 IC50 = 653 nM T63816 CVZ64I 122648649 IC50 > 1000 nM T63816 CW03VD 126582837 IC50 = 68.15 nM T63816 C5UV6J 126582839 IC50 = 32.05 nM T63816 CR9AC4 126582841 IC50 = 120.03 nM T63816 C1HS3A 126582843 IC50 = 23.42 nM T63816 CFI58L 126582907 IC50 = 132.88 nM T63816 CMT02Y 126582908 IC50 > 10000 nM T63816 CE4CI8 127025178 IC50 > 10000 nM T63816 CM38EU 127025541 IC50 = 10000 nM T63816 CA14VM 127027506 IC50 = 2092.35 nM T63816 CB9PL5 127027507 IC50 > 10000 nM T63816 CBOJ07 127027508 IC50 > 10000 nM T63816 CT18SH 127027509 IC50 > 10000 nM T63816 CG8NU7 127027995 IC50 > 10000 nM T63816 CMJ25Z 127028836 IC50 = 730 nM T63816 CP3L7U 127028844 IC50 = 150 nM T63816 CV07OM 127028943 IC50 > 10000 nM T63816 CV9I8D 127030313 IC50 = 17100 nM T63816 CB8HR2 129104138 IC50 > 50000 nM T63816 CCH65A 129104183 IC50 > 50000 nM T63816 CFH8Q4 129104227 IC50 > 50000 nM T63816 C6HM5P 129104349 IC50 > 50000 nM T63816 CZTF90 129104374 IC50 > 50000 nM T63816 CUJ2P5 129104402 IC50 > 50000 nM T63816 CY3I6X 129104426 IC50 = 29000 nM T63816 C8IEV4 130258911 IC50 = 1445 nM T63816 C6X3HG 132145728 IC50 = 4817 nM T63816 C8O9DP 132157820 IC50 = 4438 nM T63816 C4KE3N 132938351 IC50 = 7120 nM T63816 C05FVT 134492522 IC50 > 10000 nM T63816 C14FWK 135348858 IC50 = 19500 nM T63816 CS1V6A 135367138 IC50 > 50000 nM T63816 CVO59N 135367789 IC50 > 50000 nM T63816 CDY18W 135407493 IC50 > 100000 nM T63816 CW2I4R 135412048 IC50 > 100000 nM T63816 C7U0AV 135412194 IC50 > 100000 nM T63816 CI28ZH 135424818 IC50 = 358 nM T63816 CS54TL 135437514 IC50 > 100000 nM T63816 C36MUC 135441620 IC50 > 100000 nM T63816 CRB8M1 135444536 IC50 > 100000 nM T63816 CX5D6J 135446479 IC50 = 32500 nM T63816 C1TOK2 135449197 IC50 > 100000 nM T63816 CW25GL 135462117 IC50 > 100000 nM T63816 CCL28F 135473106 IC50 > 100000 nM T63816 CYA60G 135497781 IC50 > 100000 nM T63816 C01EZF 135567459 IC50 = 44000 nM T63816 CU0TV8 135589922 IC50 = 0.002 ug.mL-1 T63816 CRQ95S 135771947 IC50 = 0.001 ug.mL-1 T63816 CGB67N 135869606 IC50 = 125000 nM T63816 C8X5LO 135928012 Ki = 950 nM T63816 CI2YE8 135928628 IC50 > 100000 nM T63816 C50NIS 136025837 IC50 > 100000 nM T63816 C4OS0V 136025842 IC50 > 100000 nM T63816 CX7Z5B 136025843 IC50 > 100000 nM T63816 CB8EM9 136025984 IC50 > 100000 nM T63816 C49MUG 136025986 IC50 > 100000 nM T63816 C0OLS8 136030779 IC50 = 30000 nM T63816 CIA7R4 136030780 IC50 > 100000 nM T63816 C24LKN 136030781 IC50 > 100000 nM T63816 CH7Y3C 136086920 IC50 > 100000 nM T63816 C3VDL5 136086921 IC50 > 100000 nM T63816 C9GOB5 136086922 IC50 > 100000 nM T63816 CE3ZL7 136086923 IC50 > 100000 nM T63816 CJZ5F3 136086924 IC50 = 54200 nM T63816 CT19ND 136110961 IC50 > 100000 nM T63816 CY9U0E 136173089 IC50 > 50000 nM T63816 C32MPU 136173094 IC50 > 50000 nM T63816 CRPN39 136645466 IC50 > 10000 nM T63816 C67EFJ 137628684 IC50 > 1000 nM T63816 CP0BN3 137631704 Ki > 50000 nM T63816 C31MPL 137631726 IC50 > 10000 nM T63816 CPOF51 137632251 Ki > 50000 nM T63816 C84MIY 137633138 IC50 > 100000 nM T63816 C73PDL 137634086 IC50 > 100000 nM T63816 CZ1FK2 137635119 IC50 > 50000 nM T63816 CAWZ25 137635575 IC50 > 100 nM T63816 CK1S0F 137637029 IC50 = 25 nM T63816 CTUL07 137638741 IC50 > 100 nM T63816 C69IOZ 137639088 IC50 > 10000 nM T63816 C5QC2N 137643440 IC50 > 10000 nM T63816 CGMN16 137647616 Ki > 50000 nM T63816 CM65KH 137647813 IC50 > 100 nM T63816 C2RHM6 137647860 IC50 = 447 nM T63816 CDXE54 137649646 Ki > 50000 nM T63816 C5FHD3 137652442 IC50 = 500 nM T63816 CB15PI 137652670 Ki > 50000 nM T63816 C1SBN5 137654946 IC50 = 1980 nM T63816 CI6R3W 137656303 Ki > 50000 nM T63816 C76OGQ 137656942 IC50 > 30000 nM T63816 C5BM7T 137657586 IC50 > 100000 nM T63816 C1DL3P 137657892 Ki > 50000 nM T63816 C8D2GT 137658785 Ki > 50000 nM T63816 CAQ62X 137701235 Ki = 3400 nM T63816 CA3C4O 138454792 IC50 > 1000 nM T63816 CN2UH1 139303146 IC50 > 20000 nM T63816 C7XI0V 141764754 IC50 = 473 nM T63816 CX0E9B 142505968 IC50 = 100000 nM T63816 CKBF56 142506033 IC50 = 70910 nM T63816 CLND62 142506170 IC50 = 100000 nM T63816 CGNQ74 142506189 IC50 = 1751 nM T63816 C1T3IQ 142506210 IC50 = 11290 nM T63816 CP5HF8 142506225 IC50 = 1428 nM T63816 C1EF9X 145950102 IC50 = 98.8 nM T63816 CRKM19 145950884 IC50 = 12000 nM T63816 CV3QO5 145951170 IC50 > 10000 nM T63816 CFE4G6 145952135 IC50 = 198 nM T63816 CKG98W 145953085 IC50 > 100000 nM T63816 CM53ZB 145954785 IC50 = 117000 nM T63816 CGP9X1 145955496 IC50 = 180 nM T63816 C9IV1C 145959866 IC50 > 10000 nM T63816 CK1XI0 145960971 IC50 > 10000 nM T63816 C1X5EO 145962694 IC50 = 21000 nM T63816 C2XS8E 145968675 IC50 > 100000 nM T63816 CP53JS 145977717 IC50 > 10000 nM T63816 CW6US1 145981665 IC50 > 10000 nM T63816 CWD0A9 145983712 Ki > 10000 nM T63816 C56MWZ 145986208 Ki > 10000 nM T63816 C0GMR1 146585718 IC50 = 381 nM T63816 C0YXS8 147254231 IC50 = 5611 nM T63816 CN71OS 149405396 IC50 = 16180 nM T63816 C8S3MF 150076000 IC50 > 300 nM T63816 C9FIY4 153534005 IC50 > 10000 nM T63816 CIG6K4 155510915 IC50 = 11000 nM T63816 CQ5BL7 155512551 IC50 = 8100 nM T63816 CJ8IQ0 155513281 IC50 = 2 nM T63816 CRTJ01 155513435 IC50 = 31 nM T63816 CE4H7I 155513471 IC50 > 50000 nM T63816 CW3VT9 155514603 IC50 = 11000 nM T63816 CZ84WI 155515284 IC50 = 14000 nM T63816 CUKG21 155515602 IC50 > 50000 nM T63816 CYJ53T 155515864 IC50 = 2200 nM T63816 CA1J3N 155517086 IC50 > 100000 nM T63816 CL72ME 155517175 IC50 > 10000 nM T63816 CY54TU 155518062 IC50 = 600 nM T63816 CEH2N5 155518106 IC50 > 100000 nM T63816 CAD06U 155519254 IC50 = 3530 nM T63816 CDY5H6 155519645 IC50 > 10000 nM T63816 CYAC34 155519955 IC50 = 33 nM T63816 C3MX5D 155520119 IC50 = 9400 nM T63816 CZ75FW 155521272 IC50 = 27000 nM T63816 CP67LK 155523130 IC50 = 3000 nM T63816 C1POL9 155523278 IC50 = 103 nM T63816 C6KIO8 155523903 IC50 = 25 nM T63816 CAE1B9 155525509 IC50 = 22 nM T63816 CN7B1T 155525782 IC50 > 100000 nM T63816 C71UNO 155527385 Ki = 9540 nM T63816 CAR39I 155528228 IC50 = 22 nM T63816 CZ70PO 155529066 IC50 > 50000 nM T63816 C49NGT 155529137 IC50 > 50000 nM T63816 C9L6OC 155529247 IC50 = 972 nM T63816 CN3W5J 155531452 IC50 = 21000 nM T63816 CK2UY4 155531957 IC50 = 3800 nM T63816 C02GPA 155531979 IC50 = 6 nM T63816 C8Y9AI 155533604 IC50 = 119 nM T63816 CIZ46A 155533876 IC50 > 30000 nM T63816 CF69UC 155534005 IC50 > 50000 nM T63816 C6LB5D 155535084 IC50 > 30000 nM T63816 CO1L9U 155535427 IC50 = 22 nM T63816 C2JH0S 155537112 IC50 > 10000 nM T63816 CTF98X 155537473 IC50 > 10000 nM T63816 CAG9P4 155537573 IC50 = 17000 nM T63816 CTU3X6 155538087 IC50 > 50000 nM T63816 CLD19W 155539311 IC50 > 10000 nM T63816 CU6V4Q 155539319 IC50 > 50000 nM T63816 C6U0FM 155540189 IC50 = 1400 nM T63816 CN7E6U 155542755 IC50 > 50000 nM T63816 CP4L1F 155544459 IC50 = 5100 nM T63816 CXR86J 155545078 IC50 = 16000 nM T63816 CF2O4J 155546325 IC50 > 50000 nM T63816 CS3GO2 155546558 IC50 = 5500 nM T63816 C8XP0N 155546580 IC50 = 55 nM T63816 C0AU1L 155546632 IC50 = 20000 nM T63816 C1D4PI 155547606 Ki = 25200 nM T63816 C7Q8WO 155547936 IC50 = 30 nM T63816 C90FBZ 155549087 IC50 > 50000 nM T63816 C4Z5JX 155550827 IC50 = 32000 nM T63816 CE01AP 155551891 IC50 = 3.4 nM T63816 C05ZVG 155552130 IC50 = 11100 nM T63816 C76FVO 155552531 IC50 = 25 nM T63816 CF19RE 155554004 IC50 = 40 nM T63816 CGDF76 155554360 IC50 > 30000 nM T63816 CXGE59 155554383 IC50 = 26 nM T63816 CT7GW1 155555345 IC50 = 2700 nM T63816 CE5P4I 155555900 IC50 = 18 nM T63816 C7QTU1 155555957 IC50 = 8800 nM T63816 CV71PJ 155557724 IC50 = 57 nM T63816 CC62UI 155559872 IC50 > 10000 nM T63816 C3RX4V 155561731 IC50 = 25 nM T63816 CGL24S 155562249 IC50 = 6800 nM T63816 CU5M1Y 155563135 IC50 = 49 nM T63816 CPNA06 155564750 IC50 > 50000 nM T63816 CZDC03 155565491 IC50 > 30000 nM T63816 CG65CR 155565674 IC50 = 4100 nM T63816 CD05RS 155566122 IC50 = 20000 nM T63816 C4A0RK 155566461 IC50 > 50000 nM T63816 C51BFK 155566644 IC50 > 10000 nM T63816 C04CGS 155567444 IC50 > 50000 nM T63816 CS03PJ 155568350 IC50 > 50000 nM T63816 C46XEM 155568884 IC50 = 18 nM T63816 D00GBB 11449246 Ki = 20 nM T63816 D00KFF 9882812 Ki = 5.1 nM T63816 D00XTC 44437872 IC50 = 25 nM T63816 D01DOV 23634888 IC50 = 31200 nM T63816 D01YBR 44591988 IC50 = 16100 nM T63816 D02HVH 11427204 IC50 = 32 nM T63816 D02NAF 44437870 IC50 = 2.4 nM T63816 D02NVY 44437869 IC50 = 1.6 nM T63816 D02NWS 279980 IC50 = 140000 nM T63816 D02VVU 44328873 EC50 = 5000 nM T63816 D03BQS 45482666 IC50 = 2320 nM T63816 D03PRG 44437878 IC50 = 2.7 nM T63816 D03QOD 239512 IC50 = 250 nM T63816 D04CDZ 44437873 IC50 = 70 nM T63816 D04KQF 6675804 Ki = 9124.2 nM T63816 D04UVL 1133083 IC50 > 50000 nM T63816 D05OVV 11993691 IC50 = 1300 nM T63816 D06IMY 44626296 IC50 = 250 nM T63816 D07MYE 5355635 IC50 = 19460 nM T63816 D09RKA 72946782 IC50 > 1000 nM T63816 D0A4HF 45482630 IC50 = 700 nM T63816 D0E0TA 44454650 IC50 > 50000 nM T63816 D0E8UH 44437879 IC50 = 1.6 nM T63816 D0E9DD 16095101 IC50 = 2280 nM T63816 D0FN5D 45482672 IC50 = 1100 nM T63816 D0G1EX 44437876 IC50 = 56 nM T63816 D0H4YW 3611 Ki > 20000 nM T63816 D0I4RK 45482660 IC50 = 4500 nM T63816 D0K7QR 45269423 IC50 = 220 nM T63816 D0M1ZI 16095112 IC50 = 3660 nM T63816 D0M9LJ 44454415 IC50 > 50000 nM T63816 D0MD7H 44454143 IC50 > 50000 nM T63816 D0N5RV 44437875 IC50 = 4.2 nM T63816 D0N9AK 44138031 IC50 = 38800 nM T63816 D0PK9V 45482643 IC50 = 960 nM T63816 D0Q2GM 44454416 IC50 > 50000 nM T63816 D0Q5DI 71462653 Ki = 7570 nM T63816 D0Q5MC 24753719 IC50 > 100000 nM T63816 D0Q9PO 16095114 IC50 = 3160 nM T63816 D0R3XO 44437883 IC50 = 5.2 nM T63816 D0R7JA 53344908 Ki = 90.5 nM T63816 D0T0SK 44138032 IC50 = 2040 nM T63816 D0T4JQ 264 IC50 > 2000000 nM T63816 D0U0EZ 44437880 IC50 = 4 nM T63816 D0U8FC 759408 IC50 > 50000 nM T63816 D0W1PV 6918328 IC50 = 1 nM T63816 D0X4QC 44437877 IC50 = 3.2 nM T63816 D0Z6HR 44437874 IC50 = 2.2 nM T63816 D0Z6MI 44437868 IC50 = 1.8 nM T63816 D0Z8PX 24757913 IC50 = 3000 nM T09128 D0J3SU 9847835 Ki = 4000 nM T09128 D0LD9S 1103 EC50 = 8500 nM T09128 CF0PY8 25378 EC50 = 50000 nM T09128 C8JFN3 31239 EC50 = 21000 nM T09128 C2FQZ5 2318649 EC50 = 50000 nM T09128 C0DJ3A 2870452 EC50 = 25000 nM T09128 CMPI31 2882842 EC50 = 25000 nM T09128 CQ9K2E 3614377 EC50 = 66000 nM T09128 CO58XD 5311161 IC50 > 100000 nM T09128 C1KR5B 5327301 Ki = 30000 nM T09128 C37TKL 5327302 Ki = 9000 nM T09128 C64ZMN 5327304 Ki = 960 nM T09128 C3IZ2W 5327307 Ki = 16000 nM T09128 C16DTL 5327308 Ki = 21000 nM T09128 C4O3QY 5327309 Ki = 64000 nM T09128 C3GUM7 5327310 Ki = 37000 nM T09128 CFN2P6 9800285 Ki = 6500 nM T09128 C4XO3K 9821545 Ki = 4900 nM T09128 C6S3KT 9840223 Ki > 25000 nM T09128 CX67SZ 10826725 Ki > 25000 nM T09128 CDX7A4 10963183 Ki = 30000 nM T09128 CDT9G3 11467504 IC50 > 10 nM T09128 C3USR9 11543714 IC50 = 530 nM T09128 C17OJS 11572844 IC50 = 859 nM T09128 C6UAV3 11632008 IC50 = 233 nM T09128 C91JNO 11639020 IC50 = 231 nM T09128 C4MCW2 11646889 IC50 = 537 nM T09128 CH20JE 11652994 IC50 = 5670 nM T09128 CD8WB9 44304162 Ki = 11000 nM T09128 C8D5TB 44364680 Ki = 11000 nM T09128 C7RX9I 44418960 Ki = 29000 nM T09128 CDY2W5 49796910 IC50 > 10 nM T09128 CE8T0H 54597799 IC50 = 50 nM T09128 CFD30Q 56659222 IC50 = 41 nM T09128 CM64OW 56659923 IC50 = 86 nM T09128 C1NMH3 56659924 IC50 = 2260 nM T09128 CUD26P 56663392 IC50 = 413 nM T09128 CS3B4M 56663393 IC50 = 150 nM T09128 C8TZ9N 56666800 IC50 = 573 nM T09128 CHW0D3 56666820 IC50 = 32000 nM T09128 CZO8E4 56666821 IC50 = 52800 nM T09128 COZ26R 56669572 IC50 = 1334 nM T09128 C4J3TX 56670225 IC50 = 1980 nM T09128 C0BKU5 56670226 IC50 = 163 nM T09128 CD4QG1 56670255 IC50 = 772 nM T09128 CH3Y9M 56670256 IC50 = 219 nM T09128 CF38EO 56673751 IC50 = 2190 nM T09128 CW1R2X 56677088 IC50 = 50000 nM T09128 C8DN0E 56677089 IC50 = 136 nM T09128 C8MYW9 56679735 IC50 = 635 nM T09128 C8X7AY 56680385 IC50 = 6670 nM T09128 CB2R1I 56680416 IC50 = 1600 nM T09128 C72RGY 56683063 IC50 = 108 nM T09128 CKU26O 56683064 IC50 = 246 nM T09128 C1U8MW 56683723 IC50 = 459 nM T09128 C3FCG0 56683745 IC50 = 5533 nM T09128 CGY3W2 71471109 IC50 > 100000 nM T09128 CANH70 71716242 IC50 = 13100 nM T09128 C40WIR 71718085 IC50 > 100000 nM T09128 CU75VK 71719897 IC50 > 100000 nM T09128 CBV6F1 71720507 IC50 > 100000 nM T09128 C9QKI3 127020966 IC50 > 100000 nM T09128 CU42CE 155567829 IC50 > 100000 nM T09128 D0N5MU 4117381 Ki > 50000 nM T09128 D0Q9XX 515950 Ki > 50000 nM T09128 D0V6DX 10640 IC50 = 1530 nM T09128 D0Y5IQ 44255320 IC50 = 5000 nM T80513 D0F1LZ 176 EC50 = 12000 nM T80513 D0I7IB 5222465 EC50 = 10100 nM T80513 CC80OM 651809 EC50 = 1096.48 nM T80513 CZN6S9 743974 EC50 > 31622.78 nM T80513 C7GFP2 3142521 EC50 = 6760.83 nM T80513 CMIX24 3142523 EC50 = 1202.26 nM T80513 C7AGR5 3142525 EC50 = 1348.96 nM T80513 CMHQ78 3144722 EC50 = 3630.78 nM T80513 CXU07I 3144726 EC50 = 1621.81 nM T80513 CN0FQ9 11610220 EC50 = 537.03 nM T80513 CV8GA4 11646235 EC50 = 524.81 nM T80513 CZ7U2W 46869922 EC50 > 10000 nM T80513 C6NIF3 67072752 EC50 > 10000 nM T80513 CA24JF 86803193 EC50 > 10000 nM T80513 CNQ59Y 86803224 EC50 > 10000 nM T80513 CNW92C 91885415 EC50 = 128.82 nM T80513 CXKQ09 122184686 EC50 > 10000 nM T80513 C6OPM1 127048827 EC50 > 10000 nM T80513 CH9S7P 127048842 EC50 > 10000 nM T80513 C6V3FP 127050770 EC50 > 10000 nM T80513 CE94RI 127051658 EC50 > 10000 nM T80513 C7GX3P 129743659 EC50 = 1230.27 nM T80513 CPBG95 134136959 EC50 > 10000 nM T80513 CJ30RW 134141489 EC50 > 10000 nM T80513 CY3ZF0 134146590 EC50 > 10000 nM T80513 CAG0Y1 134151150 EC50 > 10000 nM T80513 C7MF0A 137633536 EC50 > 50000 nM T80513 CBG58K 137659266 EC50 > 10000 nM T80513 COG0M1 155511466 EC50 = 144.54 nM T80513 CK69YZ 155513981 EC50 = 1000 nM T80513 CQA3G9 155514154 EC50 < 100000 nM T80513 CB3JT2 155514597 EC50 = 645.65 nM T80513 C70XLO 155514799 EC50 = 3548.13 nM T80513 C6U9DV 155516172 EC50 = 251.19 nM T80513 CF9C7T 155516295 EC50 = 724.44 nM T80513 C3NS6Z 155516418 EC50 = 1659.59 nM T80513 C7GWC9 155518116 EC50 = 2818.38 nM T80513 CXMQ29 155518312 EC50 = 5495.41 nM T80513 C08WJD 155519653 EC50 = 501.19 nM T80513 CYZR43 155521449 EC50 = 1071.52 nM T80513 C9C5LB 155522979 EC50 = 707.95 nM T80513 C7PR9T 155526048 EC50 = 691.83 nM T80513 C6N9RK 155528851 EC50 = 3388.44 nM T80513 CXA7M9 155532033 EC50 = 10471.29 nM T80513 C2GZF8 155534056 EC50 = 1584.89 nM T80513 C8VYZ6 155534079 EC50 = 524.81 nM T80513 CZA3K4 155534383 EC50 = 1778.28 nM T80513 CDZ95Q 155534708 EC50 = 616.6 nM T80513 CX2NY4 155535071 EC50 = 1380.38 nM T80513 C4P6KC 155535425 EC50 = 11220.18 nM T80513 CKQ87B 155536193 EC50 = 354.81 nM T80513 CVSZ29 155536391 EC50 = 4897.79 nM T80513 C9TC1Q 155538299 EC50 = 1096.48 nM T80513 CWB5Y6 155538420 EC50 = 7762.47 nM T80513 CY1TZ8 155539179 EC50 = 288.4 nM T80513 CH2V8J 155539478 EC50 = 691.83 nM T80513 C3GI6P 155540026 EC50 = 35481.34 nM T80513 CG7XH4 155540222 EC50 = 398.11 nM T80513 C60DUL 155544770 EC50 = 371.54 nM T80513 C34SZG 155546001 EC50 = 162.18 nM T80513 CC35LX 155551702 EC50 = 5495.41 nM T80513 CV97NX 155553095 EC50 = 691.83 nM T80513 CI3C0Z 155553285 EC50 = 245.47 nM T80513 C9ST1J 155553549 EC50 = 602.56 nM T80513 CX0GY1 155558278 EC50 = 3890.45 nM T80513 C6MF1Z 155558623 EC50 = 380.19 nM T80513 CH3D6C 155560731 EC50 = 588.84 nM T80513 CG9X8Y 155560774 EC50 = 190.55 nM T80513 C2P8CS 155561259 EC50 = 251.19 nM T80513 CC7NQ5 155561832 EC50 = 263.03 nM T80513 CD96CN 155565387 EC50 = 1949.84 nM T80513 CCI7Q1 155569134 EC50 = 870.96 nM T80513 D07FPQ 81326 EC50 = 22387.21 nM T80513 D08ZYC 11595431 EC50 < 50118.72 nM T80513 D0S5BG 1032 EC50 = 10715.19 nM T80513 D0T4JQ 264 EC50 = 12000 nM T63484 D00VZZ 92786 IC50 = 66000 nM T63484 D0B4RU 8955 IC50 = 81400 nM T63484 D0K0EK 5881 Ki = 6200 nM T63484 D0H5HO 5879 IC50 > 200000 nM T63484 D0O8FW 441302 Ki = 3000 nM T63484 D0F7WQ 71613 IC50 = 20800 nM T63484 CU86PZ 92787 IC50 = 4300 nM T63484 CRV48L 101789 IC50 = 15800 nM T63484 C01PMJ 101927 IC50 > 200000 nM T63484 CK8I2F 102030 IC50 = 15800 nM T63484 CL6YM7 247020 IC50 = 5300 nM T63484 CNZG68 256280 IC50 = 47000 nM T63484 C8UX5A 6010075 IC50 > 80000 nM T63484 C5WVC8 9799337 IC50 = 48000 nM T63484 C0V4FO 11426281 IC50 > 200000 nM T63484 CJGI15 11695962 IC50 = 6300 nM T63484 CJ1DN0 11870468 IC50 > 200000 nM T63484 CPJ86G 11877475 IC50 = 900 nM T63484 CWV17O 14828758 IC50 = 128000 nM T63484 CB5G9A 15481096 IC50 > 200000 nM T63484 CZ5C6E 20054822 IC50 = 5200 nM T63484 C9ALM3 24792850 IC50 > 80000 nM T63484 CN3L7F 44542342 IC50 > 200000 nM T63484 CE01UH 46373715 IC50 > 80000 nM T63484 CQ73AJ 46374338 IC50 > 80000 nM T63484 C7SQD0 53362047 IC50 > 80000 nM T63484 CTF4Q0 53362048 IC50 > 80000 nM T63484 CDY7L4 53362050 IC50 > 80000 nM T63484 CZQU68 53362052 IC50 > 80000 nM T63484 CG2KY9 53362055 IC50 > 80000 nM T63484 C0YSU5 53362059 IC50 > 80000 nM T63484 CQGC50 53362065 IC50 > 80000 nM T63484 CG2F0U 53362067 IC50 > 80000 nM T63484 C03POB 53362068 IC50 > 80000 nM T63484 CBC9E1 53362070 IC50 > 80000 nM T63484 CLC2Z0 53362072 IC50 > 80000 nM T63484 C6EAF9 53362073 IC50 > 80000 nM T63484 CPD29J 53377471 IC50 > 80000 nM T63484 C61VDQ 53377474 IC50 > 80000 nM T63484 C4RPO2 53389323 IC50 > 80000 nM T63484 CG83RE 53389324 IC50 > 80000 nM T63484 CSVU32 53389325 IC50 > 80000 nM T63484 CP46LF 53481934 IC50 > 80000 nM T63484 CC1N3B 53481936 IC50 > 80000 nM T63484 CHFD01 53481937 IC50 > 80000 nM T63484 C46ADU 53481938 IC50 > 80000 nM T63484 CE9IS4 53481941 IC50 > 80000 nM T63484 C17GQR 53481943 IC50 > 80000 nM T63484 C6BVZ4 53495059 IC50 > 80000 nM T63484 CVGX16 56639562 IC50 > 80000 nM T63484 CWJ39B 57521581 IC50 > 200000 nM T63484 CNW40L 57521582 IC50 > 200000 nM T63484 C32UWT 57521583 IC50 > 200000 nM T63484 CM3O7W 57521584 IC50 = 5000 nM T63484 C81AOQ 57521685 IC50 = 12200 nM T63484 CP6A8T 57521686 IC50 = 1000 nM T63484 CENR56 57521687 IC50 = 1700 nM T63484 CC75TG 57521688 IC50 > 200000 nM T63484 CKF89I 57521689 IC50 = 7800 nM T63484 CM8JA4 57521690 IC50 = 6600 nM T63484 C3JSC1 57521797 IC50 = 70500 nM T63484 CC4U3T 57521798 IC50 = 9900 nM T63484 C63CNG 57521799 IC50 = 1200 nM T63484 CHV4J1 57521800 IC50 > 200000 nM T63484 CD4YJ6 57521801 IC50 > 200000 nM T63484 CS52MX 57521802 IC50 > 100000 nM T63484 CZG6J9 57521901 IC50 > 200000 nM T63484 CIE9T3 57521902 IC50 > 200000 nM T63484 CAU50J 57521903 IC50 = 3400 nM T63484 C9LD3I 57521904 IC50 = 11000 nM T63484 C0VM3L 57521905 IC50 = 20300 nM T63484 CF47GZ 57521906 IC50 = 2000 nM T63484 CE9HL7 57522025 IC50 = 37800 nM T63484 CQ5NB3 57522027 IC50 > 200000 nM T63484 CR64LU 57522028 IC50 > 200000 nM T63484 CLVH41 57522029 IC50 > 200000 nM T63484 CME40I 57522030 IC50 > 200000 nM T63484 C32LDG 57522031 IC50 = 34900 nM T63484 CBZ67A 57522140 IC50 = 41600 nM T63484 CDE1M6 57522141 IC50 = 3800 nM T63484 C7V9LT 57522142 IC50 = 1200 nM T63484 CD1OG8 70084189 IC50 > 200000 nM T63484 CL2J1A 70684225 IC50 = 9300 nM T63484 CBSR19 70684226 IC50 = 2500 nM T63484 C0GW7J 70690523 IC50 > 200000 nM T63484 C1LCN4 71449852 IC50 > 80000 nM T63484 C6J2NR 71449853 IC50 > 80000 nM T63484 C5Z4CE 71449854 IC50 > 80000 nM T63484 C18LQC 71449855 IC50 > 80000 nM T63484 CTE6Q3 71451667 IC50 > 80000 nM T63484 CFWN57 71453501 IC50 > 80000 nM T63484 CE37BN 71453502 IC50 > 80000 nM T63484 CC3H4S 71455212 IC50 > 80000 nM T63484 CZP3K0 71455213 IC50 > 80000 nM T63484 C0AB7Z 71457004 IC50 > 80000 nM T63484 CJ15US 71457005 IC50 > 80000 nM T63484 CRED95 71457006 IC50 > 80000 nM T63484 C86UYD 71460678 IC50 > 80000 nM T63484 CQ8L7U 71460679 IC50 > 80000 nM T63484 CB59WQ 71460680 IC50 > 80000 nM T63484 CMS83Z 71460681 IC50 > 80000 nM T63484 CJ2OK1 145950768 Ki > 2000000 nM T63484 CVF87I 145952051 Ki = 22300 nM T63484 CT0I8W 145953919 Ki > 200000 nM T63484 C8S3PB 145955700 Ki = 129000 nM T63484 C1EJY6 145957987 Ki = 16800 nM T63484 CF94AT 145958182 Ki = 35400 nM T63484 CSI93L 145958583 Ki > 400000 nM T63484 CH31ZG 145958859 Ki > 200000 nM T63484 CLOJ01 145959704 Ki > 200000 nM T63484 D03PBN 101771 IC50 = 31600 nM T62265 C7ROK9 2817700 IC50 = 840 nM T62265 C7A2HT 4614391 IC50 > 100000 nM T62265 C6L4BC 36575534 IC50 > 100000 nM T62265 C0SZ3E 56350379 IC50 > 100000 nM T62265 C1ZC8A 112526404 IC50 > 100000 nM T62265 C95MFW 146014943 IC50 = 62 nM T62265 CW46RX 155510397 IC50 > 100000 nM T62265 COY8Z3 155510513 IC50 = 92 nM T62265 CC62VI 155510884 IC50 > 100000 nM T62265 CFPX70 155513608 IC50 = 11000 nM T62265 C3CDP7 155515711 IC50 = 430 nM T62265 C0NL8G 155518027 IC50 = 99000 nM T62265 C8Z9OP 155525037 IC50 > 100000 nM T62265 CEXB27 155529213 IC50 = 120 nM T62265 C8CZL0 155534381 IC50 = 2300 nM T62265 CL84DR 155535556 IC50 > 100000 nM T62265 CG21ND 155542073 IC50 > 100000 nM T62265 CEUV65 155558032 IC50 = 22000 nM T62265 CQC46X 155563015 IC50 = 5400 nM T62265 CN06KC 155563467 IC50 = 42000 nM T62265 D08PKS 448393 IC50 = 140 nM T82720 D05ADP 160355 IC50 = 1200 nM T82720 D09JEJ 24748573 IC50 = 6.4 nM T82720 D0E3TC 44259 IC50 = 0.967 nM T82720 D00OWF 5280953 IC50 = 28 nM T82720 D05BVP 3232621 IC50 = 697 nM T82720 D08DIJ 71529610 IC50 = 0.28 nM T82720 D09CDR 77105816 IC50 = 34 nM T82720 D0CC7E 77105818 IC50 = 42 nM T82720 D0DT5I 71529599 IC50 = 2.83 nM T82720 D0JQ0Z 46916176 IC50 = 83 nM T82720 D0NS6I 10037501 IC50 = 4100 nM T82720 D0PJ1W 71529622 IC50 = 1.07 nM T82720 D0PO8N 117881270 IC50 = 157 nM T82720 D0Q3VZ 135398522 IC50 = 44 nM T82720 CVMO57 95875 IC50 > 10000 nM T82720 C3D1HC 762415 IC50 = 3800 nM T82720 CFA92X 1237489 IC50 = 5800 nM T82720 CD1A9T 1241605 IC50 = 1500 nM T82720 CU80LI 3233012 IC50 = 452 nM T82720 CW4C3P 3235048 IC50 > 10000 nM T82720 CLM7V5 5371900 IC50 > 10000 nM T82720 CO6KI2 5930298 IC50 = 2630 nM T82720 C69ZOB 10453611 IC50 = 43 nM T82720 CP04JC 11666231 IC50 = 60 nM T82720 CPI54D 11953235 IC50 = 15 nM T82720 CJ0NW4 12235681 IC50 = 100 nM T82720 CR3BS0 12248905 IC50 = 260 nM T82720 CX27EP 13975510 IC50 = 10500 nM T82720 C5VPH9 16129448 IC50 = 1530 nM T82720 CMW42V 19079253 IC50 = 5200 nM T82720 C48UIA 21413325 IC50 = 710 nM T82720 CW2YQ0 25141335 IC50 = 6400 nM T82720 CGLQ20 44223952 IC50 = 1510 nM T82720 CR6VH2 44223953 IC50 = 506 nM T82720 C2IBW0 44223954 IC50 = 2271 nM T82720 CS3Q2Y 44223955 IC50 = 458 nM T82720 C5M1UN 44223957 IC50 = 1441 nM T82720 CK8G1T 44223965 IC50 = 130 nM T82720 CJ8KD4 44223966 IC50 = 846 nM T82720 CCW0V4 44223967 IC50 = 1125 nM T82720 CF78WD 44223968 IC50 > 10000 nM T82720 CNE30X 44223970 IC50 = 25 nM T82720 CYR45S 44223971 IC50 = 180 nM T82720 CLZ62P 44223973 IC50 = 73 nM T82720 CIXB09 44223974 IC50 = 431 nM T82720 C2OBX8 44223977 IC50 = 938 nM T82720 C3JBN1 44968184 IC50 = 1781 nM T82720 CYW79D 44968186 IC50 = 231 nM T82720 C5OYK3 44968199 IC50 = 4269 nM T82720 C2T0EM 44968221 IC50 = 7990 nM T82720 C8NA2J 44968224 IC50 = 304 nM T82720 CR8DC5 44968225 IC50 = 4036 nM T82720 CV19YK 44968230 IC50 = 352 nM T82720 CD4ZN1 44968231 IC50 = 4420 nM T82720 CQ0ZI7 45141513 IC50 = 20000 nM T82720 C16QFN 46172966 IC50 > 10000 nM T82720 CB32ET 46172972 IC50 = 6782 nM T82720 CN26HW 46172980 IC50 = 411 nM T82720 CGH05O 46172984 IC50 = 871 nM T82720 C4X1BO 46316704 IC50 = 300 nM T82720 C15EJK 46916169 IC50 = 4927 nM T82720 CHG8C4 46916170 IC50 = 446 nM T82720 CI56BA 46916172 IC50 = 48 nM T82720 CZ5DJ4 46916177 IC50 = 534 nM T82720 CXK37B 46916178 IC50 = 734 nM T82720 CL1GW0 46916179 IC50 = 313 nM T82720 CZ6DK4 46916182 IC50 = 856 nM T82720 CCUG10 46926515 IC50 = 137 nM T82720 C9NC6W 46926516 IC50 = 18 nM T82720 CZ1D2A 46926518 IC50 = 12 nM T82720 C7S6HT 46926519 IC50 = 55 nM T82720 CG1K5A 46926520 IC50 > 10000 nM T82720 CVF48X 46926521 IC50 = 42 nM T82720 C4ULH5 46926522 IC50 = 18 nM T82720 CPE98Z 46926523 IC50 = 38 nM T82720 C6WLX1 46926524 IC50 = 8862 nM T82720 C61LUI 46926526 IC50 = 884 nM T82720 C0IVD1 46926527 IC50 = 112 nM T82720 CE4SU5 47298428 IC50 = 300 nM T82720 CAYI59 49795862 IC50 = 599 nM T82720 C1UQN4 49795863 IC50 = 514 nM T82720 CU8OC0 49795864 IC50 = 829 nM T82720 C7T5HW 49795865 IC50 = 93 nM T82720 C6N8EY 49795866 IC50 = 125 nM T82720 C7XS1Z 49795867 IC50 = 179 nM T82720 C5EWG8 49855158 IC50 = 240 nM T82720 CS6N8Z 54581884 IC50 = 333 nM T82720 C3UC1Q 56929347 IC50 = 370 nM T82720 CDK93W 56946894 IC50 = 40 nM T82720 C3MFV7 57414126 IC50 = 18.3 nM T82720 CR3I5F 57418686 IC50 = 1700 nM T82720 CPK49W 57523834 IC50 = 2970 nM T82720 CWB05Y 57523919 IC50 = 68 nM T82720 CW1CM5 57523921 IC50 = 96 nM T82720 C7K9YV 57523922 IC50 = 40 nM T82720 CB5MW8 57524010 IC50 = 586 nM T82720 C8N9SO 57524101 IC50 = 135 nM T82720 C45GPV 57524102 IC50 = 9 nM T82720 C6Z9FB 57524195 IC50 = 13 nM T82720 C91BAE 57524196 IC50 = 248 nM T82720 CPK6C8 57524269 IC50 = 11 nM T82720 C2XEQ5 57524335 IC50 = 75 nM T82720 CK2DM8 57524410 IC50 = 233 nM T82720 CJ91XM 57524491 IC50 < 5 nM T82720 C4O0QZ 57524820 IC50 = 252 nM T82720 CTID23 57524821 IC50 = 134 nM T82720 C3KRE2 57524829 IC50 = 774 nM T82720 CQM73T 57524896 IC50 = 48 nM T82720 CFH12N 57524901 IC50 = 17 nM T82720 C4WGF1 57524903 IC50 = 1150 nM T82720 CVTB94 58047131 IC50 = 1600 nM T82720 CF6K1Y 58857683 IC50 = 9100 nM T82720 C56MAG 59379853 IC50 = 820 nM T82720 CIS84M 60162923 IC50 = 560 nM T82720 C37NKO 67129970 IC50 = 5020 nM T82720 CK80LJ 67130050 IC50 > 10000 nM T82720 CV63UL 67240318 IC50 > 10000 nM T82720 CKY3W6 68108530 IC50 = 1005 nM T82720 CYW71X 68108891 IC50 = 26 nM T82720 COPZ25 68108932 IC50 = 31 nM T82720 C9VMR0 68109014 IC50 = 18 nM T82720 C6PE0H 68109248 IC50 = 101 nM T82720 C0COB2 68109381 IC50 = 615 nM T82720 CB8SP0 68109626 IC50 = 21 nM T82720 C7GRV2 68755406 IC50 > 10000 nM T82720 COL1Q7 70370469 IC50 = 1894 nM T82720 CQA3B0 70370554 IC50 = 8 nM T82720 CCM6X2 71272330 IC50 = 7.7 nM T82720 C5JHE3 71277785 IC50 = 31.5 nM T82720 COB76S 71529590 IC50 = 485.8 nM T82720 CY30GN 71529591 IC50 = 11.13 nM T82720 C4OP6Q 71529598 IC50 = 3.48 nM T82720 CA8T4S 71529600 IC50 = 9.64 nM T82720 CW9CI7 71529601 IC50 = 71.98 nM T82720 C70TAN 71529603 IC50 = 7.69 nM T82720 C4IS7N 71529612 IC50 = 93.84 nM T82720 C9UTB3 71529613 IC50 = 18.78 nM T82720 C5OPK8 71529614 IC50 = 64.28 nM T82720 C1RP0Y 71529624 IC50 = 25.21 nM T82720 CQ4GS7 71529626 IC50 = 7.72 nM T82720 CG5EZ4 71529627 IC50 = 37.34 nM T82720 CW63BV 71529753 IC50 = 19.22 nM T82720 CPQU78 71529756 IC50 = 4.2 nM T82720 C3VAQ2 71608036 IC50 = 6.55 nM T82720 CBY80T 72716071 IC50 = 3 nM T82720 CAQ87R 72724765 IC50 > 10000 nM T82720 CB1EX4 72724904 IC50 > 10000 nM T82720 C36SAZ 72725030 IC50 > 10000 nM T82720 C0T6IK 73345875 IC50 = 1.63 nM T82720 CD6G8Z 73347380 IC50 = 0.59 nM T82720 C4BV9L 73426232 IC50 > 1000 nM T82720 C21JAS 76853169 IC50 = 910 nM T82720 CU04XY 77105624 IC50 = 100 nM T82720 CTIA65 77105820 IC50 = 900 nM T82720 CKB1P9 77106023 IC50 = 28 nM T82720 CXYW85 77106025 IC50 = 300 nM T82720 C2UDS0 77106026 IC50 > 10000 nM T82720 C97SJD 77106027 IC50 = 460 nM T82720 CFQ10R 77106028 IC50 = 220 nM T82720 CO14DP 77106030 IC50 = 590 nM T82720 C9G3PA 77106234 IC50 = 220 nM T82720 CPD27I 77106235 IC50 = 1100 nM T82720 CLOR37 77106236 IC50 = 93 nM T82720 C2GLD8 77106237 IC50 = 160 nM T82720 C0GYK1 86765296 IC50 = 350 nM T82720 C4BKA6 89429109 IC50 > 10000 nM T82720 C2FOK4 89494280 IC50 = 2100 nM T82720 CE5L8V 90388565 IC50 = 1200 nM T82720 CWE9I2 91664021 IC50 = 600 nM T82720 CW58AE 91664022 IC50 = 4900 nM T82720 CB25UZ 91664023 IC50 = 1400 nM T82720 CB5GU0 91668530 IC50 = 140 nM T82720 C8G5IT 118714396 IC50 = 200 nM T82720 CB8G1T 118714397 IC50 = 6100 nM T82720 CTUZ03 118714399 IC50 = 2700 nM T82720 CRV8H7 118714400 IC50 = 800 nM T82720 C7PAU6 118714401 IC50 = 1300 nM T82720 C6FQ8M 118714402 IC50 = 200 nM T82720 CXK5C3 118714403 IC50 = 7000 nM T82720 CJ89SC 118714404 IC50 = 400 nM T82720 C1GU9B 118714405 IC50 = 400 nM T82720 CF2IE6 118714406 IC50 = 2300 nM T82720 C2ZBH0 118714407 IC50 = 1000 nM T82720 CK64OD 118714410 IC50 = 2300 nM T82720 CP27TX 118735321 IC50 = 85 nM T82720 CJH0M1 118735322 IC50 = 2 nM T82720 CA7Z4X 118735323 IC50 = 1 nM T82720 C76XKT 118735324 IC50 = 16 nM T82720 CI26FD 118735325 IC50 = 34 nM T82720 CU8T1C 118735326 IC50 = 9 nM T82720 C1PDE5 118735327 IC50 = 4 nM T82720 CQ0GS4 118735328 IC50 = 4 nM T82720 C3KLT1 118735329 IC50 = 5 nM T82720 C1RAP6 118735330 IC50 = 168 nM T82720 CQ45PF 118735331 IC50 = 25 nM T82720 C56MYE 118735332 IC50 = 98 nM T82720 CP26VF 118735333 IC50 = 898 nM T82720 CSR3N8 118735334 IC50 = 810 nM T82720 C3TS7H 118735335 IC50 = 2118 nM T82720 C4DQ5K 118735336 IC50 = 192 nM T82720 C4DQX9 118735337 IC50 = 3069 nM T82720 CBY4K3 118735338 IC50 = 7 nM T82720 C5CK7W 118735339 IC50 = 3 nM T82720 CO83PN 122181013 IC50 = 210 nM T82720 C69ULZ 122181014 IC50 = 80 nM T82720 CIG8Y1 122181016 IC50 = 3000 nM T82720 CRJS41 122181017 IC50 = 1000 nM T82720 CVB03H 122181018 IC50 = 230 nM T82720 C6SJ3X 122181019 IC50 > 10000 nM T82720 C7L5PG 122181021 IC50 > 10000 nM T82720 C58CJI 122181022 IC50 > 10000 nM T82720 CC2G8N 122181024 IC50 = 1900 nM T82720 CV5BQ9 122181097 IC50 = 1300 nM T82720 C5KB1C 122184057 IC50 = 70 nM T82720 CVBF01 127030212 IC50 = 2640 nM T82720 CI93ZA 127030213 IC50 = 4290 nM T82720 C8LQV4 127030516 IC50 = 1680 nM T82720 CS12RU 127031435 IC50 = 70 nM T82720 CZXP62 127031750 IC50 = 6700 nM T82720 C3E5YO 127032014 IC50 = 1050 nM T82720 C2ZD8S 127032024 IC50 = 900 nM T82720 CXWY73 127032324 IC50 = 2170 nM T82720 C2LWZ1 129318964 IC50 = 690 nM T82720 C4W6AD 129897084 IC50 = 206 nM T82720 CM8DK3 134813913 IC50 = 110 nM T82720 CPCA46 135566559 IC50 = 37 nM T82720 CBU0J4 135604653 IC50 > 10000 nM T82720 CH0Q2Z 136234577 IC50 = 110 nM T82720 CV6F4N 136234578 IC50 = 72 nM T82720 C2G3JY 136234579 IC50 > 10000 nM T82720 C1TGM4 136244455 IC50 = 11 nM T82720 CLF3B0 136259623 IC50 = 5.68 nM T82720 CJC89A 136333957 IC50 = 78.6 nM T82720 CCAZ26 137631656 IC50 = 80 nM T82720 C3QAV9 137631819 IC50 = 1700 nM T82720 CI43OC 137632412 IC50 = 51 nM T82720 CG8Y0U 137633419 IC50 = 13000 nM T82720 CH4PN9 137633814 IC50 = 17 nM T82720 CS9TU2 137633985 IC50 > 10000 nM T82720 CI1E8V 137634241 IC50 > 10000 nM T82720 C83UKG 137634382 IC50 = 220 nM T82720 CNT7S3 137634818 IC50 > 10000 nM T82720 CCP7X5 137635304 IC50 = 3600 nM T82720 C1AK8X 137635556 IC50 = 3600 nM T82720 CV7OF5 137635713 IC50 = 1900 nM T82720 C5QWE1 137635926 IC50 = 38 nM T82720 CKZF46 137638065 IC50 = 3500 nM T82720 CRV1E4 137638175 IC50 > 1000 nM T82720 CCX37E 137638472 IC50 = 140 nM T82720 CPO87L 137638509 IC50 = 37 nM T82720 C1UI5N 137638944 IC50 = 1200 nM T82720 CH4RP3 137639514 IC50 = 520 nM T82720 CX3MQ1 137639546 IC50 = 110 nM T82720 CH3S8N 137640038 IC50 = 170 nM T82720 CXM4G7 137640811 IC50 = 130 nM T82720 CF83TG 137640934 IC50 = 180 nM T82720 CRSQ71 137641785 IC50 = 42 nM T82720 CWVE69 137643514 IC50 = 1400 nM T82720 CYA1F7 137643721 IC50 = 90 nM T82720 C2AG3W 137643887 IC50 = 28000 nM T82720 C4DS3I 137643955 IC50 = 1800 nM T82720 C75MLQ 137643957 IC50 = 130 nM T82720 CWIP72 137644498 IC50 = 960 nM T82720 CZ4U0W 137644802 IC50 = 190 nM T82720 CPJ42V 137644974 IC50 > 10000 nM T82720 C8VTQ9 137645650 IC50 = 2200 nM T82720 C7ZOV3 137645947 IC50 > 10000 nM T82720 CL5NX9 137646497 IC50 = 2100 nM T82720 CJ5O2Q 137646673 IC50 = 4100 nM T82720 CK6S5T 137646758 IC50 > 1000 nM T82720 COU37W 137647335 IC50 = 110 nM T82720 CMI2H3 137647526 IC50 = 83 nM T82720 C7O2AW 137647969 IC50 > 10000 nM T82720 CNW13G 137648784 IC50 = 128 nM T82720 CGK5P2 137649037 IC50 = 198 nM T82720 C5OJH2 137649318 IC50 = 680 nM T82720 C9IO5F 137649821 IC50 = 38 nM T82720 C9QNG8 137650421 IC50 = 7200 nM T82720 CWG94C 137650926 IC50 = 4600 nM T82720 C8MKN0 137651314 IC50 = 1200 nM T82720 CKL0P4 137651538 IC50 = 3600 nM T82720 CJ14XO 137651668 IC50 = 3800 nM T82720 CH6L2T 137652047 IC50 = 1100 nM T82720 C2B5CY 137652970 IC50 = 1200 nM T82720 C48DVU 137653000 IC50 = 130 nM T82720 C01URE 137653446 IC50 = 1100 nM T82720 CDX83M 137654129 IC50 = 32 nM T82720 C47FBV 137654225 IC50 = 1200 nM T82720 CX7V6P 137654671 IC50 > 1000 nM T82720 C7IU4J 137655848 IC50 = 53 nM T82720 CQEJ60 137656868 IC50 = 32 nM T82720 C3Y2CR 137657691 IC50 = 172 nM T82720 CA10CX 137657812 IC50 = 138 nM T82720 C39SEV 137658150 IC50 = 1100 nM T82720 CX8YL9 137658187 IC50 = 51 nM T82720 CX4M8T 137658722 IC50 > 1000 nM T82720 CA2PY1 137658970 IC50 = 410 nM T82720 CJ1TB2 137659239 IC50 = 1800 nM T82720 C3U2OB 137659350 IC50 = 510 nM T82720 C7MI2G 137661183 IC50 > 10000 nM T82720 CIX41F 137661315 IC50 = 7100 nM T82720 CD0FV8 137661355 IC50 = 3400 nM T82720 C9HPG8 137661516 IC50 = 330 nM T82720 C9BAN7 140682661 IC50 = 24.1 nM T82720 CENA85 145979136 IC50 = 138 nM T82720 C2B7VE 145979242 IC50 = 154.3 nM T82720 CNFH75 145979518 IC50 = 130 nM T82720 C2OF0R 145980649 IC50 = 326.3 nM T82720 C53HBS 145981791 IC50 = 13.8 nM T82720 CXD83F 145985653 IC50 = 130 nM T82720 CFYE93 145986392 IC50 = 131.7 nM T82720 CTWD68 145988875 IC50 = 383 nM T82720 CWP60I 145989404 IC50 = 67.1 nM T82720 C0BW5M 145990753 IC50 = 298.5 nM T82720 C1MUA8 145991360 IC50 = 98.8 nM T82720 CPK48V 145991505 IC50 = 251.4 nM T82720 CZU8J6 145992124 IC50 = 72.9 nM T82720 CK56CB 145993150 IC50 = 1513 nM T82720 CQ48WH 145993525 IC50 = 218.8 nM T82720 C5YW8Q 145993622 IC50 = 8 nM T82720 C2MD1Q 155513187 IC50 > 10000 nM T82720 D00AQR 71529770 IC50 = 4.74 nM T82720 D06CXU 46926513 IC50 = 7 nM T82720 D08NQM 5289247 IC50 = 80 nM T82720 D0UI7U 46926514 IC50 = 1156 nM T82720 D0X9PI 71529752 IC50 = 0.24 nM T30420 CIBX58 6604934 IC50 = 700 nM T30420 C5N3LG 44251522 IC50 > 40000 nM T30420 C70VHB 53315882 IC50 > 10000 nM T30420 CA8LQ7 53711055 EC50 < 1000 nM T30420 C4XJ5N 78357767 IC50 = 7300 nM T30420 COH4I6 101882828 IC50 > 250000 nM T30420 CO8R1D 101882829 IC50 = 52000 nM T30420 C1GRM5 101882830 IC50 = 9500 nM T30420 CRNH89 101882831 IC50 = 61000 nM T30420 CMNF08 101882832 IC50 = 46000 nM T30420 C3IC2P 101882833 IC50 = 11000 nM T30420 CXYV89 101882834 IC50 = 7900 nM T30420 C2W9QU 101882835 IC50 = 48000 nM T30420 CO07HF 101882836 IC50 > 250000 nM T30420 C6K7QZ 101882837 IC50 = 130000 nM T30420 C61CHJ 101882839 IC50 = 8000 nM T30420 CWHP38 101882840 IC50 = 40000 nM T30420 C6BNV7 101882841 IC50 = 8700 nM T30420 CDI62N 118708786 Ki = 2000 nM T30420 CT43XM 118708787 IC50 = 67000 nM T30420 CI3J5M 118708788 IC50 = 36000 nM T30420 C2W1AN 118708789 IC50 = 43000 nM T30420 CSPO31 118708790 IC50 = 7900 nM T30420 CL4K9S 118708791 IC50 = 7900 nM T30420 C9HN8K 118708792 IC50 = 21000 nM T30420 CFS36T 118708793 IC50 = 35000 nM T30420 CV2AX9 118708794 IC50 = 32000 nM T30420 C9ASR5 118708795 IC50 = 29000 nM T30420 CD36JB 118708796 IC50 = 25000 nM T30420 C4UO3M 118708797 IC50 = 34000 nM T30420 CD8OT5 118708798 IC50 = 58000 nM T30420 CT5Z6S 118708799 IC50 > 250000 nM T30420 CPT0Y2 118708800 IC50 = 94000 nM T30420 C1C6PZ 118708801 IC50 > 250000 nM T30420 CWI4U6 118708802 IC50 = 9200 nM T30420 CIGL09 118708803 IC50 > 250000 nM T30420 C2NPB5 118708804 IC50 > 250000 nM T30420 CV1W9F 118708805 IC50 = 37000 nM T30420 C0SK1A 118708806 IC50 = 37000 nM T30420 CS19MI 118708807 IC50 > 250000 nM T30420 CN0J5M 118708808 IC50 > 250000 nM T30420 C3WUZ5 118708809 IC50 > 250000 nM T30420 CH0W6T 122191350 IC50 = 24000 nM T30420 CTHS62 122191351 IC50 > 250000 nM T30420 CHM2U9 122191691 IC50 = 26000 nM T30420 CH5C8G 122191692 IC50 = 40000 nM T30420 CYL64J 122191693 IC50 = 40000 nM T30420 CEJ2T1 122191694 IC50 = 43000 nM T30420 C5L0MX 122191695 IC50 > 250000 nM T30420 CQ2K9O 122191696 IC50 > 250000 nM T30420 C4HTQ2 122191697 IC50 = 63000 nM T30420 C4JLO6 122191698 IC50 > 250000 nM T30420 COJ01Q 122191699 IC50 > 250000 nM T30420 CO0U3X 122191700 IC50 = 110000 nM T30420 CV3NM6 122191701 IC50 = 15000 nM T30420 CP9A4S 122191702 IC50 > 250000 nM T30420 CY7TH6 122191703 IC50 > 250000 nM T30420 CE2GM3 122191704 IC50 > 250000 nM T30420 CP6G2J 122191705 IC50 > 250000 nM T30420 CW64FT 122191706 IC50 > 250000 nM T30420 C79XZG 122191707 IC50 > 250000 nM T30420 C19OFM 122191708 IC50 > 250000 nM T30420 CZ6ED1 122191709 IC50 > 250000 nM T30420 C42GRW 122191710 IC50 > 250000 nM T30420 CD95KS 122191711 IC50 > 250000 nM T30420 CH64ED 122191712 IC50 > 250000 nM T30420 CH2QV3 122191713 IC50 > 250000 nM T30420 CHZ80X 122191714 IC50 > 250000 nM T30420 CZ64PU 122191715 IC50 > 250000 nM T30420 C4NT2G 122191716 IC50 > 250000 nM T30420 CB68XY 134149139 Ki = 50 nM T30420 C3IUY4 136845639 IC50 > 250000 nM T30420 CZ8EC6 155540557 IC50 > 200000 nM T30420 CAE87C 155557235 IC50 > 200000 nM T30420 CN2B8J 155560229 IC50 = 39000 nM T30420 D07HPE 481747 IC50 = 500 nM T30420 D0CX4W 46901937 IC50 > 40000 nM T99818 D02OZE 2724385 IC50 = 290 nM T99818 CFEQ05 16120562 IC50 = 340 nM T99818 C1K4QJ 16121811 IC50 = 570 nM T99818 CTI1C6 122182551 IC50 = 11000 nM T99818 C1YV8G 122363019 IC50 = 9800 nM T60514 CU6ON8 9802264 IC50 = 7600 nM T60514 C6HZB8 11531111 IC50 = 53500 nM T60514 CRJT72 76308593 IC50 = 86800 nM T60514 C3BUD9 76312290 IC50 = 9000 nM T60514 D0B3WX 5475158 IC50 = 35000 nM T97592 D02RJY 11442891 Ki = 61 nM T97592 D02XNW 5494449 IC50 = 4.6 nM T97592 D0A1AQ 5329099 IC50 = 210 nM T97592 D0CY1B 6420138 IC50 = 65 nM T97592 D0E3TC 44259 IC50 = 2.42 nM T97592 D0EJ3B 24856041 IC50 = 1 nM T97592 D0IQ0Z 46885626 Ki = 1.5 nM T97592 D0J6AB 24748204 IC50 = 12 nM T97592 D0Q7RE 16007391 Ki = 17 nM T97592 C7PEG0 10200408 Ki = 11 nM T97592 CK6U2S 11249084 IC50 = 120 nM T97592 C1UFM0 11497983 IC50 = 17 nM T97592 CACS26 11561968 Ki > 1000 nM T97592 CU0E8O 11690457 Ki > 10000 nM T97592 CB0AP2 11705863 Ki > 1000 nM T97592 C9JT4S 11847343 IC50 = 62 nM T97592 C8FLH6 16202152 IC50 = 227 nM T97592 CL81VC 21100709 IC50 = 4750 nM T97592 CX18GT 46889932 IC50 = 19 nM T97592 CV4X7L 49787166 IC50 = 3 nM T97592 CCSP59 49800150 IC50 = 1950 nM T97592 CD2K4R 50908681 Ki > 1000000 nM T97592 CT3EW2 59292007 IC50 > 1000 nM T97592 COH62U 60097413 IC50 > 5000 nM T97592 C1MR8Q 60097495 IC50 > 2000 nM T97592 CV63UL 67240318 IC50 > 10000 nM T97592 C4Q6FE 71815105 IC50 = 67.2 nM T97592 CJ2T9E 76332983 IC50 = 259 nM T97592 C2IN3C 118710236 IC50 = 153.5 nM T97592 CO8Z2N 129900111 IC50 = 53 nM T97592 CIP61L 134153498 IC50 = 63 nM T97592 CJ65LQ 135423783 IC50 > 100000 nM T97592 C2WL8M 135423784 IC50 > 100000 nM T97592 CNKD13 135423790 IC50 = 1000 nM T97592 C48NWF 135423791 IC50 = 900 nM T97592 CEVL69 135423792 IC50 = 700 nM T97592 C6HGC3 135423793 IC50 = 600 nM T97592 C1W6EI 135423851 IC50 > 100000 nM T97592 CYH51Q 135423852 IC50 > 100000 nM T97592 C21PTY 136104462 IC50 > 100000 nM T97592 C7XO8B 136104463 IC50 > 100000 nM T97592 C7UH8T 136104464 IC50 = 28000 nM T97592 C7R2PD 136104467 IC50 > 100000 nM T97592 CLEN23 136104468 IC50 > 100000 nM T97592 CWLJ05 136104469 IC50 > 100000 nM T97592 C8C5XL 145984893 IC50 = 3 nM T97592 C2MD1Q 155513187 IC50 > 10000 nM T97592 C13GYL 127031746 IC50 < 5000 nM T97592 D00UTU 136104465 IC50 = 4500 nM T97592 D06AGN 136043837 IC50 = 700 nM T97592 D07ADX 54764565 IC50 = 290 nM T97592 D0CE3R 5312137 IC50 = 17 nM T97592 D0I1IK 136104466 IC50 = 1000 nM T97592 D0V6LP 136043836 IC50 = 400 nM T97592 D0Y0ES 3707 IC50 = 300 nM T19433 D06TNL 3278 IC50 = 122300 nM T19433 D0E6OC 5282230 IC50 = 11600 nM T19433 CU16EY 5345 IC50 = 27000 nM T19433 CL60FN 40854 IC50 > 300000 nM T19433 CI6CG7 67262 IC50 = 9200 nM T19433 C5S3EK 77812 IC50 = 105000 nM T19433 CN8PG3 93177 IC50 = 220000 nM T19433 C12FXI 121026 IC50 = 890000 nM T19433 CM5Q1T 230783 IC50 = 12400 nM T19433 CC5DI9 695906 IC50 = 138 nM T19433 C12DHB 767167 IC50 = 33000 nM T19433 CRC5J0 786892 IC50 = 45000 nM T19433 CL64UQ 2742128 IC50 = 26400 nM T19433 CF9G8H 2763788 IC50 = 23 nM T19433 CUQR43 2767324 IC50 = 3800 nM T19433 CU5T0L 2805912 IC50 = 34700 nM T19433 CC86NQ 2814179 IC50 < 1 nM T19433 C0ZHD3 4412670 IC50 = 17400 nM T19433 C72YAC 5062655 IC50 = 6270 nM T19433 CF4U5P 15402200 IC50 = 13000 nM T19433 CFJC05 16665631 IC50 = 23 nM T19433 CMI84P 16665941 IC50 = 9.5 nM T19433 C9LIR6 17897432 IC50 = 5000 nM T19433 C9M8ZU 22030791 IC50 = 8900 nM T19433 C35KJQ 24764436 IC50 = 920 nM T19433 CZ8O7V 24776309 IC50 = 994 nM T19433 CE1A9T 24776311 IC50 = 75 nM T19433 CUD02I 24776312 IC50 = 1500 nM T19433 C1XQD8 24991044 EC50 = 35 nM T19433 C2L6MB 25099474 IC50 = 7 nM T19433 C7C2UY 39038262 IC50 = 8500 nM T19433 CO16MN 42571591 IC50 = 170 nM T19433 CIG35E 46899922 IC50 = 700 nM T19433 CBC8T7 46899923 IC50 = 1900 nM T19433 CQY4X8 46899924 IC50 = 19900 nM T19433 C8OY9E 46899925 IC50 = 10800 nM T19433 CNK21I 46899926 IC50 = 10800 nM T19433 C52EBC 46900085 IC50 = 43800 nM T19433 CNI80S 46900086 IC50 = 1800 nM T19433 CSHD27 46900087 IC50 = 57900 nM T19433 COV2L3 46900088 IC50 = 8000 nM T19433 C27XVK 46900089 IC50 = 7100 nM T19433 CMEV83 46900244 IC50 = 72500 nM T19433 C9Q5CK 46900245 IC50 = 5070 nM T19433 C1YC8L 46900246 IC50 = 88500 nM T19433 C0YQ8T 46900247 IC50 = 91000 nM T19433 CWM21I 46900248 IC50 = 57600 nM T19433 CVL63N 46900249 IC50 = 53300 nM T19433 CB0F4O 46900397 IC50 = 24600 nM T19433 CBP18V 46900398 IC50 = 14700 nM T19433 CHKU85 46900399 IC50 = 24800 nM T19433 C04TBO 46900400 IC50 = 20500 nM T19433 CK6WS7 46900401 IC50 = 38000 nM T19433 CI9O8G 46900402 IC50 = 54000 nM T19433 C84XNE 46900403 IC50 = 1200 nM T19433 CO76CD 49864074 IC50 = 25900 nM T19433 C18QGS 49864099 IC50 = 3700 nM T19433 C23ESD 49864100 IC50 = 1300 nM T19433 CQ8K0U 49864134 IC50 = 23000 nM T19433 CPI07G 51210626 IC50 = 6900 nM T19433 C0ASE2 56962331 IC50 = 845 nM T19433 CYI4Q0 56962332 IC50 = 8.26 nM T19433 C8MA2Z 57383478 IC50 = 2.34 nM T19433 CZS54E 58316756 IC50 = 500 nM T19433 CYRL52 59200016 IC50 = 6 nM T19433 CIS96H 59200042 IC50 = 3 nM T19433 C3N5WJ 59673077 IC50 = 274 nM T19433 CY5ZS3 59743886 IC50 = 0.2 nM T19433 C9MW6P 59743926 EC50 = 130 nM T19433 CH0J7A 60167934 IC50 < 10 nM T19433 C32CTA 60196237 IC50 = 1480 nM T19433 CV48ZU 70692285 IC50 = 662 nM T19433 C1R2OU 70694357 IC50 = 280 nM T19433 C58PBX 71720415 IC50 > 10000 nM T19433 CING05 76322208 IC50 = 40 nM T19433 CYJP12 76336683 IC50 = 17000 nM T19433 CW36LE 91799244 IC50 = 180 nM T19433 C0IE1M 110489845 IC50 = 7700 nM T19433 C4JT9K 110489888 IC50 = 3100 nM T19433 CWF29K 110489892 IC50 = 1600 nM T19433 CGR42J 110489893 IC50 > 50000 nM T19433 CX47ZE 110489903 IC50 = 870 nM T19433 CZ7BR1 110489918 IC50 = 2400 nM T19433 CWP3R6 110489926 IC50 = 200 nM T19433 CYOQ04 118736784 IC50 = 70 nM T19433 CYX37P 118736785 EC50 = 350 nM T19433 CTO09D 118736786 IC50 = 26 nM T19433 CE45PM 118736787 IC50 = 32 nM T19433 CY7C3S 118736788 IC50 = 35 nM T19433 CK9F2M 118736789 IC50 = 43 nM T19433 CA89HU 118736790 IC50 = 130 nM T19433 C1P2KJ 118736791 IC50 = 1200 nM T19433 CI6TO0 118736792 IC50 = 31 nM T19433 C0ZLB4 118736793 IC50 = 48 nM T19433 C81SZP 118736794 IC50 = 230 nM T19433 C1VQC8 118736796 IC50 = 320 nM T19433 C0JXG2 118736798 IC50 = 590 nM T19433 C38CKS 129247272 IC50 = 14 nM T19433 CME4A3 129247298 IC50 = 52 nM T19433 C05NGH 129247316 IC50 = 120 nM T19433 CG3ML2 129247320 IC50 = 26 nM T19433 C5UEW1 129247333 IC50 = 230 nM T19433 CF16NB 129247350 IC50 = 280 nM T19433 CILC96 129247356 IC50 = 8.2 nM T19433 CEO8X2 129247382 IC50 = 98 nM T19433 CNV07D 129247462 IC50 = 20 nM T19433 CFL3A7 129247606 IC50 = 9.9 nM T19433 C7WS4G 129274871 IC50 = 25 nM T19433 CD0LH1 129276274 IC50 = 56 nM T19433 CGYC12 145983882 IC50 = 8 nM T19433 CGQ53M 145985449 IC50 = 10 nM T19433 C5TP4M 155511296 IC50 = 57 nM T19433 CS19YX 155513454 IC50 = 100 nM T19433 CI23UJ 155514356 IC50 = 1200 nM T19433 CWT57K 155514556 IC50 = 4100 nM T19433 C9NB5Q 155516371 IC50 = 17 nM T19433 CL4V3X 155516451 IC50 = 2200 nM T19433 CA97QE 155518468 IC50 = 110 nM T19433 C0IQ6H 155520357 IC50 = 1400 nM T19433 CLUE26 155522629 IC50 = 9.7 nM T19433 CMS37F 155524220 IC50 = 49 nM T19433 C1R3NO 155527379 IC50 = 1400 nM T19433 C4TEP6 155528204 IC50 = 640 nM T19433 C2FG9Y 155528603 IC50 = 220 nM T19433 C0MCN6 155532559 IC50 = 23 nM T19433 C9G0QW 155532574 IC50 = 7800 nM T19433 CVU5P2 155533035 IC50 = 530 nM T19433 CR7QI2 155533894 IC50 = 320 nM T19433 C5OTM0 155538303 IC50 = 120 nM T19433 C1KW2M 155538467 IC50 = 73 nM T19433 C0OGM8 155538781 IC50 = 340 nM T19433 C0LSW2 155542115 IC50 = 250 nM T19433 C6PM9N 155542799 IC50 = 350 nM T19433 CBE75S 155542838 IC50 = 6900 nM T19433 C47PKV 155543877 IC50 = 170 nM T19433 C5FUA1 155544194 IC50 = 15 nM T19433 CV1R8F 155544242 IC50 = 1800 nM T19433 C2XSD3 155546004 IC50 = 16 nM T19433 CD2W5V 155550171 IC50 = 160 nM T19433 C7I3SP 155550421 IC50 = 420 nM T19433 C02EYC 155551492 IC50 = 15000 nM T19433 CS7FO0 155551494 IC50 = 2300 nM T19433 C7U3BR 155552285 IC50 = 71 nM T19433 C6AN2F 155553456 IC50 = 390 nM T19433 CX0I5J 155553534 IC50 = 360 nM T19433 C2THB1 155555025 IC50 = 8500 nM T19433 C0IJ1M 155555573 IC50 = 1400 nM T19433 CIV5A3 155555774 IC50 = 590 nM T19433 C1BQ9P 155557287 IC50 = 220 nM T19433 COV3Z8 155559395 IC50 = 520 nM T19433 C28AVC 155559677 IC50 = 57 nM T19433 CPAN81 155560038 IC50 = 1400 nM T19433 CCUY89 155562545 IC50 = 250 nM T19433 CM3FR7 155563576 IC50 = 78 nM T19433 C3E7PH 155564317 IC50 = 620 nM T19433 CE4N8O 155564754 IC50 = 2000 nM T19433 CLCB64 155565549 IC50 = 200 nM T19433 CU3TA2 155567236 IC50 = 630 nM T19433 C76OWN 155567313 IC50 = 4500 nM T19433 C2MOZ4 155568551 IC50 = 110 nM T19433 D01YPD 2767330 IC50 = 3800 nM T19433 D06GJP 172469 IC50 = 200 nM T19433 D0PI1C 6540277 IC50 = 73900 nM T46245 D03TFJ 5798 Ki = 150000 nM T46245 C82HDB 1467860 Ki = 1010 nM T46245 C96LQT 1467864 Ki = 780 nM T46245 CAX89D 1467867 Ki = 2610 nM T46245 C71JQH 1467870 Ki = 17800 nM T46245 C06QOP 2726661 Ki = 700 nM T46245 CF1L9O 2841348 Ki = 7700 nM T46245 CFQE57 2882201 Ki = 4480 nM T46245 CT6VF0 2910461 Ki = 1860 nM T46245 C9LI1D 2917732 Ki = 700 nM T46245 CC12GR 2918257 Ki = 4700 nM T46245 CQ4Y6A 2918952 Ki = 2680 nM T46245 C3XR1L 2929274 Ki = 2140 nM T46245 CLE7A3 2969796 Ki = 890 nM T46245 CSCK43 3585502 Ki = 1240 nM T46245 C62UFG 3692902 Ki = 13020 nM T46245 CD10EB 4178505 Ki = 2040 nM T46245 CUR6P0 4389874 Ki = 1790 nM T46245 C5Z2TE 5153417 Ki = 5670 nM T46245 C6NZJ0 5488150 IC50 = 27900 nM T46245 CVWS50 6539180 Ki = 14720 nM T46245 CQX3A4 6539181 Ki = 11300 nM T46245 C0I4NC 6539182 Ki = 3660 nM T46245 CB23WG 6539183 Ki = 2790 nM T46245 C13PEN 6539184 Ki = 2780 nM T46245 CNF9K2 6539185 Ki = 4730 nM T46245 CPH53F 6539186 Ki = 2030 nM T46245 CB08JA 6539187 Ki = 1660 nM T46245 C0VXL6 6539188 Ki = 970 nM T46245 C5YO8C 6539189 Ki = 5660 nM T46245 CONR87 6539190 Ki = 1550 nM T46245 CRM1K8 6539191 Ki = 1120 nM T46245 C67KIL 6539192 Ki = 750 nM T46245 CM5PY2 6539193 Ki = 560 nM T46245 C3F5LP 6539194 Ki = 490 nM T46245 CY28ZX 6539195 Ki = 340 nM T46245 CEO68P 6539197 Ki = 17660 nM T46245 C1BY9H 6539198 Ki = 550 nM T46245 C7M5NK 6539199 Ki = 340 nM T46245 C2JCD5 6539200 Ki = 760 nM T46245 CXVY92 6539201 Ki = 2330 nM T46245 C8SF5C 6539202 Ki = 4830 nM T46245 CPEV18 6539203 Ki = 3730 nM T46245 CQ2W9J 6539204 Ki = 3350 nM T46245 CRTG15 6539205 Ki = 1570 nM T46245 CGQ3N7 6539206 Ki = 2000 nM T46245 CDL36X 6539207 Ki = 390 nM T46245 CJ6TE8 6539208 Ki = 7340 nM T46245 C4PHZ6 6539209 Ki = 3510 nM T46245 C6OD4G 6539210 Ki = 4480 nM T46245 CT1MU5 6539211 Ki = 400 nM T46245 C7PK8U 6539212 Ki = 4880 nM T46245 CT1J8L 6539213 Ki = 7330 nM T46245 CN08BG 6539214 Ki = 2220 nM T46245 CQ8H9S 6539215 Ki = 90 nM T46245 CAH8S4 6539216 Ki = 990 nM T46245 CT6J9F 10707952 IC50 = 16800 nM T46245 C47VMY 11252738 Ki = 1530 nM T46245 CU9K5B 11492713 Ki = 1020 nM T46245 COE1U8 11595085 Ki = 1360 nM T46245 C8BK0V 11630784 Ki = 700 nM T46245 C72UXF 17374308 Ki = 4650 nM T46245 CF5P6V 19595609 IC50 = 34600 nM T46245 C9OG5V 24858983 Ki = 1090 nM T46245 CY49XU 25015755 IC50 = 162 nM T46245 CB12QE 25022550 Ki = 6.3 nM T46245 C2M3GY 25022552 Ki = 61 nM T46245 C7UO6I 25024283 Ki = 6070 nM T46245 CN5D7J 25024284 Ki = 4560 nM T46245 C7LVC9 25024285 Ki = 600 nM T46245 CRX7N4 25024286 Ki = 5260 nM T46245 CDH68G 25024480 Ki = 9670 nM T46245 CZ31OQ 25024481 IC50 = 15000 nM T46245 CAGR41 25024686 Ki = 4870 nM T46245 CK7J0H 25054713 Ki = 130 nM T46245 CI29WX 25054968 Ki = 82 nM T46245 CT02AL 25054970 Ki = 65 nM T46245 CX43VG 25055207 Ki = 253 nM T46245 CG2F1E 25055457 Ki = 1650 nM T46245 CZN29Y 25062649 Ki = 60 nM T46245 CWE7N2 44549233 Ki = 2.6 nM T46245 C68YUT 44549234 Ki = 41 nM T46245 COSQ71 44549360 Ki = 1370 nM T46245 C5IXM6 44549361 Ki = 6720 nM T46245 C4PY5O 44549362 Ki = 830 nM T46245 CFI46Y 44549363 Ki = 620 nM T46245 CR9BY6 44549630 IC50 = 24.3 nM T46245 C91DRC 45483707 Ki = 17 nM T46245 CNGL48 45483761 Ki = 300 nM T46245 CLGA01 45483789 Ki = 360 nM T46245 C4TU3P 45483790 Ki = 340 nM T46245 CBG82Q 45483791 Ki = 620 nM T46245 CHG40B 45483805 Ki = 900 nM T46245 CPW17J 45483806 Ki = 230 nM T46245 CZN03A 45483807 Ki = 18 nM T46245 CF37ZD 45483820 Ki = 39 nM T46245 CU38KM 45483826 Ki = 20 nM T46245 CPV6K5 45483832 Ki = 83 nM T46245 CQY5C2 50967174 Ki = 1040 nM T46245 CQL8N9 51030869 IC50 = 29 nM T46245 CVK1A5 53359057 Ki = 23 nM T46245 C46CKE 53378966 Ki = 250 nM T46245 CL8KB4 53378967 Ki = 106 nM T46245 CS0NL6 53379083 Ki = 139 nM T46245 CY1WJ2 53379085 Ki = 211 nM T46245 C4XL8I 53379087 Ki = 1310 nM T46245 CCJ1M8 53379088 IC50 = 24700 nM T46245 CS58XM 58433214 Ki = 638 nM T46245 CC70OD 58433225 Ki = 415 nM T46245 C39JKU 58433229 Ki = 351 nM T46245 CLIM92 58433234 Ki = 107 nM T46245 CPKW19 58433235 IC50 = 31700 nM T46245 C1Z8SH 58433244 Ki = 645 nM T46245 CVY49I 58433250 Ki = 335 nM T46245 C95URX 58433251 Ki = 536 nM T46245 CG05HQ 58433254 Ki = 167 nM T46245 CNQ9S4 58433255 Ki = 80 nM T46245 C3QCT0 58433259 Ki = 1140 nM T46245 C8SB6G 58433261 Ki = 702 nM T46245 CR8Y6H 58433266 Ki = 424 nM T46245 CE8L1T 58433268 Ki = 941 nM T46245 C15SZE 58433274 Ki = 382 nM T46245 C6UBM9 58433285 Ki = 716 nM T46245 C0CIR4 58433286 Ki = 333 nM T46245 C2PEK5 58433288 Ki = 157 nM T46245 CE8OF6 58433290 IC50 = 26900 nM T46245 CIR28Z 66839681 IC50 = 26000 nM T46245 CXTD95 71712421 IC50 = 208 nM T46245 CJR9B0 71712422 IC50 = 479 nM T46245 CUL9Y8 71712423 IC50 = 492 nM T46245 C0IA1Z 71712424 IC50 = 1070 nM T46245 CD39WT 71712425 IC50 = 58 nM T46245 C6O5JQ 71712427 IC50 = 482 nM T46245 C4Z9RJ 71712428 IC50 = 788 nM T46245 CGE97W 71712562 IC50 = 519 nM T46245 C7OZ9X 71712563 IC50 = 812 nM T46245 C3HP9X 71712565 IC50 = 1613 nM T46245 C63IZK 71712566 IC50 = 239 nM T46245 C4JGO8 71712567 IC50 = 381 nM T46245 CPZ67D 71712568 IC50 = 463 nM T46245 COQ3J6 71712569 IC50 = 711 nM T46245 CMKS70 71712714 IC50 = 461 nM T46245 CG3TN8 71712715 IC50 = 475 nM T46245 C4T5SO 71712716 IC50 = 524 nM T46245 C4N0IC 71712717 IC50 = 1070 nM T46245 C4H3WO 71712718 IC50 = 329 nM T46245 CEX92G 71712719 IC50 = 1220 nM T46245 CILE16 71712720 IC50 = 488 nM T46245 CS4Q0Z 71712721 IC50 = 453 nM T46245 CN5CP0 71712864 IC50 = 518 nM T46245 CXT5N9 71712866 IC50 = 337 nM T46245 C5GRA3 71712867 IC50 = 158 nM T46245 CTC3I1 71712868 IC50 = 293 nM T46245 CUGM73 71712869 IC50 = 768 nM T46245 C1H8AK 71713007 IC50 = 546 nM T46245 C5R1PT 71713008 IC50 = 375 nM T46245 C6CAD3 71713009 IC50 = 3050 nM T46245 CU3A4M 71713010 IC50 = 123 nM T46245 CQPY28 71714509 IC50 = 185 nM T46245 CK38HW 71714511 IC50 = 437 nM T46245 CP26XJ 71714512 IC50 = 405 nM T46245 CQX75Y 73294650 Ki = 1250 nM T46245 CTCX82 91618245 IC50 = 16.7 nM T46245 CN27US 92045043 IC50 = 4.5 nM T46245 C23LKM 125494169 IC50 = 15300 nM T46245 C1X7UR 127031185 IC50 = 15000 nM T46245 CGYT46 127032229 IC50 = 16100 nM T46245 CLEB26 127032851 IC50 = 37200 nM T46245 C5ROU4 127033256 IC50 = 14200 nM T46245 CYK6W0 127033759 IC50 = 19300 nM T46245 CO2ME5 134691747 IC50 = 500 nM T46245 CA7M9Y 134691748 IC50 = 118 nM T46245 CK6CP0 137631856 IC50 = 19.8 nM T46245 C6NX0U 137632787 IC50 = 24.7 nM T46245 C3EN1L 137632818 IC50 = 16.6 nM T46245 CQ8F7Z 137633514 IC50 = 1560 nM T46245 CM8Q6S 137633745 IC50 = 38.6 nM T46245 CPN93L 137633835 IC50 = 890 nM T46245 CY6OH4 137635128 IC50 = 1380 nM T46245 CAWC98 137635313 IC50 = 20.5 nM T46245 CNF7L5 137635503 IC50 = 9 nM T46245 CM49VJ 137635765 IC50 = 14.4 nM T46245 CIFY21 137636028 IC50 = 13.4 nM T46245 CNQ6G3 137636535 IC50 = 17.5 nM T46245 CXR19Z 137636657 IC50 = 12.5 nM T46245 CD2J6T 137637121 IC50 = 15500 nM T46245 CENK87 137637262 IC50 = 38.7 nM T46245 CZ9C1A 137637616 IC50 = 700 nM T46245 CT0EZ9 137637821 IC50 = 8.2 nM T46245 CUS9J2 137638846 IC50 = 1620 nM T46245 CD80GQ 137639416 IC50 = 3.7 nM T46245 C0UWY8 137639430 IC50 = 7.3 nM T46245 CP45JN 137639662 IC50 = 40.8 nM T46245 CPJ2S1 137639999 IC50 = 19 nM T46245 CIWR14 137640846 IC50 = 7.2 nM T46245 C9P3KJ 137640874 IC50 = 10.7 nM T46245 CK7C5T 137641146 IC50 = 3020 nM T46245 CZ76DQ 137642348 IC50 = 16.2 nM T46245 CC4FS1 137642842 IC50 = 13.8 nM T46245 CL3MB6 137643592 IC50 = 18.5 nM T46245 CQ10FI 137643681 IC50 = 6.9 nM T46245 CYNT60 137644512 IC50 = 12.5 nM T46245 C26YZE 137645120 IC50 = 2080 nM T46245 C6RG3P 137645359 IC50 = 880 nM T46245 CQ4E0B 137645555 IC50 = 7.8 nM T46245 C6J0XD 137645901 IC50 = 14.1 nM T46245 CW69EL 137645980 IC50 = 39.4 nM T46245 C4G0ZN 137646463 IC50 = 640 nM T46245 CD8XK6 137646722 IC50 = 5.3 nM T46245 CI8N6U 137647037 IC50 = 8.3 nM T46245 C5AHJ9 137648337 IC50 = 11.4 nM T46245 CEL06G 137649080 IC50 = 23.5 nM T46245 CBC60A 137649114 IC50 = 2570 nM T46245 CPR64Z 137649987 IC50 = 17.5 nM T46245 CR2I6U 137650020 IC50 = 0.7 nM T46245 CF7J5Q 137651092 IC50 = 5.5 nM T46245 CU94YO 137651162 IC50 = 830 nM T46245 CCU91X 137651629 IC50 = 5.7 nM T46245 C3MDN8 137651795 IC50 = 19.3 nM T46245 CGQ8U1 137652275 IC50 = 21.3 nM T46245 CA9GL3 137652332 IC50 = 20.2 nM T46245 CF72ML 137654220 IC50 = 4.6 nM T46245 CGW3A4 137654478 IC50 = 15.3 nM T46245 CW7B8G 137654690 IC50 = 18.4 nM T46245 C2V4OF 137654703 IC50 = 9.1 nM T46245 C85NWX 137655382 IC50 = 30.2 nM T46245 CM8Z5Q 137657425 IC50 = 41.2 nM T46245 C5D2TH 137658801 IC50 = 7.7 nM T46245 CFTQ06 137658875 IC50 = 13.8 nM T46245 CU1VT6 137659013 IC50 = 11.7 nM T46245 C4SB9N 137659404 IC50 = 940 nM T46245 C89SEL 137659624 IC50 = 790 nM T46245 C8Y2UG 137659649 IC50 = 12.3 nM T46245 CG30WB 137660255 IC50 = 4.8 nM T46245 CX2A3J 137660378 IC50 = 13 nM T46245 C9VSZ1 137661242 IC50 = 35.5 nM T46245 CZ2PS3 137661697 IC50 = 9.2 nM T46245 C3BH7W 139035065 IC50 = 6.1 nM T46245 C48PIW 145960675 IC50 = 24.7 nM T46245 CN7A6J 145960831 IC50 = 26 nM T46245 CI63HG 145960837 IC50 = 26.8 nM T46245 C60WFM 145960966 IC50 = 22 nM T46245 CLJ20S 145960977 IC50 = 7.9 nM T46245 CHDX42 145960990 IC50 = 11.4 nM T46245 C9SAO0 145961087 IC50 = 15 nM T46245 C1C4NG 145961134 IC50 = 15.8 nM T46245 C9U2OZ 145961244 IC50 = 20.6 nM T46245 C81VQO 145961291 IC50 = 15.9 nM T46245 C3TGB1 145961335 IC50 = 56.5 nM T46245 CL6MX2 145961485 IC50 = 12.9 nM T46245 CT39JY 145961797 IC50 = 15.2 nM T46245 CJLF93 145961894 IC50 = 18.4 nM T46245 CMK28W 145962056 IC50 = 7.9 nM T46245 C0ECD9 145962114 IC50 = 18.7 nM T46245 C7PC4D 145962379 IC50 = 6.4 nM T46245 CS3BO8 145962420 IC50 = 26.4 nM T46245 COQL01 145962559 IC50 = 7.9 nM T46245 CF4Y6G 145962621 IC50 = 8.8 nM T46245 C5ZLY4 145963052 IC50 = 8.8 nM T46245 CMZP17 145963175 IC50 = 11.2 nM T46245 CYT1R0 145963296 IC50 = 9 nM T46245 C82VYG 145963305 IC50 = 15 nM T46245 CS34WT 145963306 IC50 = 7.3 nM T46245 CI03MU 145963406 IC50 = 19.4 nM T46245 C6Q5SG 145963411 IC50 = 46.8 nM T46245 CIEH21 145963677 IC50 = 16.2 nM T46245 CG2T4W 145963982 IC50 = 7.5 nM T46245 CN68GB 145964168 IC50 = 48.7 nM T46245 CVJL71 145964228 IC50 = 13.4 nM T46245 C3ZMK8 145964466 IC50 = 3.6 nM T46245 C14LME 145964517 IC50 = 51 nM T46245 CM5JU2 145964518 IC50 = 12.7 nM T46245 CDC13X 145964546 IC50 = 66.8 nM T46245 C1UZ9E 145964604 IC50 = 3.8 nM T46245 CV8DL6 145965094 IC50 = 12 nM T46245 CKE03M 145966279 IC50 = 9.9 nM T46245 CR65YM 145966290 IC50 = 6.2 nM T46245 CP1YA9 145966530 IC50 = 15 nM T46245 CTP20O 145966825 IC50 = 23.5 nM T46245 CKDI27 145967192 IC50 = 89.7 nM T46245 C4Y2RH 145968476 IC50 = 17.3 nM T46245 CT49EI 145968705 IC50 = 9.4 nM T46245 CRCF38 145970051 IC50 = 11.5 nM T46245 CWTK15 145970274 IC50 = 4.5 nM T46245 C2CVY0 145972023 IC50 = 117 nM T46245 CR07XI 145972070 IC50 = 12 nM T46245 CA3JW1 145972129 IC50 = 4.8 nM T46245 CM38HG 145972134 IC50 = 17 nM T46245 CN29IT 145973024 IC50 = 8.5 nM T46245 CMZ12W 145973082 IC50 = 8.6 nM T46245 C9GM5Y 145973212 IC50 = 17.7 nM T46245 CS09XQ 145973429 IC50 = 9.9 nM T46245 CD8Z5U 145973969 IC50 = 7.8 nM T46245 CIY8E3 145974886 IC50 = 9 nM T46245 C0V3SE 145975279 IC50 = 19 nM T46245 C3J4TW 145975448 IC50 = 10.6 nM T46245 CN1T0Q 145975461 IC50 = 30.8 nM T46245 C5E6YA 145975884 IC50 = 5.5 nM T46245 CCR9L5 145976064 IC50 = 1.8 nM T46245 CG8SZ0 145976098 IC50 = 16.1 nM T46245 C1GPW4 145976241 IC50 = 16.7 nM T46245 CTR9O7 145976263 IC50 = 40.3 nM T46245 CS8BR5 145976667 IC50 = 7.7 nM T46245 C7GSU3 145977279 IC50 = 21.6 nM T46245 CUA2N3 145977317 IC50 = 7.4 nM T46245 C4RLC6 145977478 IC50 = 35.4 nM T46245 CTE08C 145977529 IC50 = 8.7 nM T46245 C9GXN7 145977704 IC50 = 53.8 nM T46245 CQ4A6Z 145978092 IC50 = 10.3 nM T46245 CCU08R 145978124 IC50 = 7 nM T46245 C5UN9J 145978632 IC50 = 15.7 nM T46245 CYK4R8 145978674 IC50 = 5.8 nM T46245 C3L6DP 155510844 IC50 = 8.6 nM T46245 C8U5JW 155511970 IC50 = 17.6 nM T46245 CE9SP5 155513434 IC50 = 23.3 nM T46245 C4JK3A 155514688 IC50 = 8.8 nM T46245 CS2K6Y 155514984 IC50 = 93 nM T46245 CIRT83 155516711 IC50 = 16.4 nM T46245 CY27QD 155517533 IC50 = 4.1 nM T46245 C7WDX3 155517834 IC50 = 1.6 nM T46245 CR1ZO2 155518173 IC50 = 30.6 nM T46245 CN0D1M 155518431 IC50 = 6.2 nM T46245 C2TJ3Z 155519633 IC50 = 3.9 nM T46245 CT8N5G 155520141 IC50 = 38.5 nM T46245 CQAG81 155520479 IC50 = 81.6 nM T46245 C57KNM 155520516 IC50 = 7.5 nM T46245 C5LRG7 155521646 IC50 = 19.4 nM T46245 CR30DT 155523348 IC50 = 13.3 nM T46245 C19JCB 155523704 IC50 = 22.9 nM T46245 C10BTO 155527363 IC50 = 4.6 nM T46245 CF1B4R 155527620 IC50 = 5.6 nM T46245 C4BGU9 155529738 IC50 = 4.7 nM T46245 CX3K1P 155530159 IC50 = 2.8 nM T46245 CAV84W 155530655 IC50 = 11 nM T46245 CS8Y3Z 155531729 IC50 = 112 nM T46245 C41BSY 155532055 IC50 = 77.5 nM T46245 CQM78C 155533886 IC50 = 32.5 nM T46245 C6XK8I 155533985 IC50 = 17.5 nM T46245 CU98NC 155534568 IC50 = 39 nM T46245 C9CD4A 155535202 IC50 = 8.2 nM T46245 C48LKZ 155535558 IC50 = 5.4 nM T46245 CBZ0L5 155537024 IC50 = 23.5 nM T46245 CEH39J 155537798 IC50 = 12.9 nM T46245 CKS4P6 155538431 IC50 = 27 nM T46245 C6J9YA 155541815 IC50 = 37.1 nM T46245 C9IX3W 155541943 IC50 = 6.8 nM T46245 C2WZA6 155542146 IC50 = 12.5 nM T46245 CG6E2N 155543281 IC50 = 1.3 nM T46245 C46SQO 155547313 IC50 = 77.3 nM T46245 CNY76A 155549691 IC50 = 15 nM T46245 C96IVL 155549874 IC50 = 3.4 nM T46245 CP79MK 155550357 IC50 = 4.5 nM T46245 C0KNO7 155552583 IC50 = 3.6 nM T46245 C2TQR4 155556105 IC50 = 78.7 nM T46245 C8WZ6J 155557554 IC50 = 69.6 nM T46245 CBS65V 155558500 IC50 = 36.9 nM T46245 C3JXV2 155558667 IC50 = 8.7 nM T46245 CC3S5V 155558712 IC50 = 53.9 nM T46245 CBXP64 155562243 IC50 = 6.5 nM T46245 C0SRL9 155562744 IC50 = 81 nM T46245 CBQ26E 155564634 IC50 = 98.8 nM T46245 C2J1WV 155564706 IC50 = 25.6 nM T46245 CP4Z1X 155564935 IC50 = 7.6 nM T46245 CWAR94 155565347 IC50 = 13.6 nM T46245 CU42JD 155566901 IC50 = 3.5 nM T46245 CX93KU 155566959 IC50 = 20.5 nM T46245 CVA58C 155567186 IC50 = 26.5 nM T46245 C10HGU 155567263 IC50 = 183 nM T46245 CDN31L 155567481 IC50 = 12.4 nM T46245 CG78XO 155567836 IC50 = 5.2 nM T46245 C9R2EB 155568709 IC50 = 25 nM T46245 D00JHN 6539196 Ki = 60 nM T46245 D0SY6C 5282073 IC50 = 45200 nM T31721 D00ENY 33032 Ki = 51 nM T31721 C9CQV1 131738 IC50 > 1000000 nM T31721 C7BKY8 164701 IC50 = 100000 nM T31721 C45TML 1755783 IC50 > 300000 nM T31721 CDK9W5 1796705 IC50 > 300000 nM T31721 C8L6JU 2177697 IC50 > 300000 nM T31721 CRQW20 2266743 IC50 > 300000 nM T31721 CO0I2U 2266913 IC50 > 300000 nM T31721 C9HE6N 2271641 IC50 > 300000 nM T31721 CH4RP6 2271698 IC50 > 300000 nM T31721 C3SL4Y 2271738 IC50 > 300000 nM T31721 C7K9MX 2283576 IC50 > 300000 nM T31721 CB6EZ4 2285406 IC50 > 300000 nM T31721 CBW36C 2287441 IC50 > 300000 nM T31721 C13DLB 2289587 IC50 > 300000 nM T31721 CZQ83G 2289624 IC50 > 300000 nM T31721 CFG35Z 2737891 IC50 > 100000 nM T31721 CYR4X2 2838960 IC50 > 100000 nM T31721 CP4L3M 2839392 IC50 > 300000 nM T31721 CF2LE3 4133412 IC50 = 8000 nM T31721 CJW9P4 5506801 IC50 > 300000 nM T31721 C5PWJ3 6505351 IC50 > 300000 nM T31721 CTBZ42 6505352 IC50 > 300000 nM T31721 C64QSY 7016554 Ki = 61659.5 nM T31721 CTMP80 9920506 Ki = 37153.52 nM T31721 C2EA8S 10219727 IC50 > 1000000 nM T31721 C53YBE 10419887 Ki > 400000 nM T31721 C2PE4O 10464763 IC50 > 1000000 nM T31721 C46KUE 10680281 Ki = 87096.36 nM T31721 C2WQB7 10877814 IC50 > 1000000 nM T31721 C83OPZ 10954230 IC50 > 1000000 nM T31721 C7Z6AX 10986716 IC50 > 1000000 nM T31721 C78YAI 10997729 IC50 > 1000000 nM T31721 CE80SU 11041159 IC50 > 1000000 nM T31721 CMSD95 11062853 IC50 > 1000000 nM T31721 C2TWR9 11063103 IC50 > 1000000 nM T31721 C0HT8M 11528550 Ki = 295120.92 nM T31721 CQ5H1B 11543205 Ki = 46000 nM T31721 C2QJU5 11616374 IC50 = 10000 nM T31721 CZ9V5S 11629898 Ki = 66069.34 nM T31721 C5E8BT 11651356 Ki = 70794.58 nM T31721 CV76LO 11667702 IC50 = 2400 nM T31721 C7SHB1 11745400 Ki = 31622.78 nM T31721 C0BM2Z 12047098 IC50 = 8400 nM T31721 C68AOJ 12047099 IC50 = 4800 nM T31721 C09XIT 12047100 IC50 = 6500 nM T31721 C1X3YB 16727662 IC50 > 300000 nM T31721 C6XLF5 24905646 Ki > 3000 nM T31721 CFI54P 24905647 Ki > 3000 nM T31721 CQK96U 24905648 Ki > 3000 nM T31721 C36NMZ 24905649 Ki = 3000 nM T31721 CB3T7C 24905650 Ki = 3000 nM T31721 C14RNW 24905651 Ki = 3000 nM T31721 CM1S2B 24905652 Ki = 1000 nM T31721 CUS45D 24905703 Ki > 3000 nM T31721 C86BUK 24905705 Ki > 3000 nM T31721 CJ25EZ 44404580 IC50 = 600 nM T31721 C0LJ8T 44404590 IC50 = 1000 nM T31721 CJD1V7 44404611 IC50 = 1000 nM T31721 CJ6ER9 44404615 IC50 = 1000 nM T31721 C4CZN1 44405320 Ki = 50118.72 nM T31721 CI94LS 44417413 Ki = 49000 nM T31721 C8TMX2 44417425 Ki = 10000 nM T31721 CR2IM7 49910175 IC50 > 300000 nM T31721 CY91US 52941382 IC50 = 117.49 nM T31721 C5ILP4 70682198 IC50 = 53000 nM T31721 C4HI0U 70789291 IC50 > 3000000 nM T31721 CP48NY 71449125 IC50 = 3000 nM T31721 C7NYC0 71449126 IC50 = 1500 nM T31721 CD03AH 71449127 IC50 = 850 nM T31721 CVST26 71450915 IC50 = 200 nM T31721 C31HCW 71450916 IC50 = 1800 nM T31721 CC15SM 71450917 IC50 = 3000 nM T31721 CBZ9D6 71450918 IC50 = 9000 nM T31721 CSO9P3 71452727 IC50 = 300 nM T31721 C23DMA 71452728 IC50 = 140 nM T31721 CE0A3V 71452729 IC50 = 5600 nM T31721 CRKN62 71452730 IC50 = 14500 nM T31721 C8X4VU 71454504 IC50 = 450 nM T31721 COUY80 71454505 IC50 = 500 nM T31721 C8QW6K 71454506 IC50 = 600 nM T31721 CKWF24 71454507 IC50 = 5000 nM T31721 CDY5K2 71456248 IC50 = 600 nM T31721 C9O7LC 71456249 IC50 = 50 nM T31721 C1HJF2 71458054 IC50 = 650 nM T31721 C3P0MQ 71461655 IC50 = 2000 nM T31721 C0P4NT 71574743 IC50 > 300000 nM T31721 CGH79X 71574744 IC50 > 300000 nM T31721 COC8W2 71574746 IC50 > 300000 nM T31721 C5U9HZ 71574747 IC50 > 300000 nM T31721 C35BOJ 71574834 IC50 > 1000000 nM T31721 CNVG02 71574836 IC50 = 100000 nM T31721 C2JS0I 71574837 IC50 > 1000000 nM T31721 CV5IT8 71574838 IC50 > 1000000 nM T31721 CL9BJ8 71574839 IC50 > 1000000 nM T31721 CCS4T2 71574840 IC50 > 1000000 nM T31721 CM5Z0I 71574841 IC50 > 300000 nM T31721 C3Z0TH 73348758 Ki = 50118.72 nM T31721 C8DGU5 90480101 IC50 > 1000000 nM T31721 CEH82V 90480134 IC50 > 1000000 nM T31721 CT2KF1 127030385 IC50 > 300000 nM T31721 CX95LC 127030386 IC50 > 300000 nM T31721 C8TS1X 127030387 IC50 > 300000 nM T31721 CF6NI8 127031290 IC50 > 300000 nM T31721 C2V5PM 132820245 IC50 = 524.81 nM T31721 CC54HS 134131748 IC50 = 100000 nM T31721 CM8O9I 134131963 IC50 = 7400 nM T31721 C26CTG 134132565 IC50 = 300000 nM T31721 CGXV98 134133631 IC50 = 3100 nM T31721 C1ZAB4 134134123 IC50 = 300000 nM T31721 CZ2WH5 134134813 IC50 = 31622.78 nM T31721 CT3MU6 134135313 IC50 = 300000 nM T31721 CTL6A4 134135682 IC50 = 75857.76 nM T31721 C0MJT1 134136786 IC50 = 150000 nM T31721 CA40DU 134137403 IC50 = 100000 nM T31721 C1L9UX 134139672 IC50 = 6456.54 nM T31721 CC24GI 134139698 IC50 > 1000000 nM T31721 CTSA19 134139982 IC50 = 10000 nM T31721 CWS62H 134140412 IC50 = 100000 nM T31721 C5QIB1 134140490 IC50 = 100000 nM T31721 CT4QN8 134141720 IC50 = 34000 nM T31721 CJF5X7 134143016 IC50 = 1000000 nM T31721 C4CT5L 134144465 IC50 = 6200 nM T31721 CL0EA9 134144947 IC50 = 150000 nM T31721 COM76W 134147363 IC50 > 300000 nM T31721 C9Q2JY 134147568 IC50 = 3000 nM T31721 CS38BI 134147884 IC50 = 12000 nM T31721 CP10YS 134148109 IC50 = 300000 nM T31721 CTPS85 134149212 IC50 = 8800 nM T31721 COP15G 134149427 IC50 = 20000 nM T31721 C6HQS8 134149488 IC50 = 1200 nM T31721 CTH41F 134149576 IC50 = 13000 nM T31721 CQ8R9N 134149841 IC50 = 63000 nM T31721 C10RSO 134150446 IC50 > 300000 nM T31721 C9N0CQ 134152035 IC50 = 300000 nM T31721 C5SN8C 134152143 IC50 = 2570.4 nM T31721 C3RAO8 134153858 IC50 = 1949.84 nM T31721 CI3HS7 134155673 IC50 = 977.24 nM T31721 CVT7Q4 134157558 IC50 = 2000 nM T31721 CHK48B 137643975 IC50 > 1000000 nM T31721 C6J8RH 137658224 IC50 > 1000000 nM T31721 CS1X0H 145952067 IC50 = 288.4 nM T31721 C2X6ST 145952092 IC50 = 2100 nM T31721 CRXG02 145952717 IC50 = 840 nM T31721 CZD62V 145953140 IC50 = 1600 nM T31721 C5SH4V 145953224 IC50 = 28000 nM T31721 C63MDC 145954707 IC50 = 128.82 nM T31721 C87HDC 145955435 IC50 = 1600 nM T31721 CT3H6G 145955563 IC50 = 870.96 nM T31721 CIN7D3 145955863 IC50 = 2691.53 nM T31721 CZ7N3B 145956590 IC50 = 2570.4 nM T31721 CFZK42 145957754 IC50 = 1174.9 nM T31721 CEX81Q 145958688 IC50 = 97000 nM T31721 C6BP3Z 145959256 IC50 = 10471.29 nM T31721 C8DIJ6 145960111 IC50 = 3090.3 nM T31721 CET93L 145971223 IC50 = 104.71 nM T31721 CGF5S1 145971489 IC50 = 30902.95 nM T31721 C30JVP 145971753 IC50 = 1202.26 nM T31721 CI04HT 145972021 IC50 = 54.95 nM T31721 C18GNB 145973375 IC50 = 94 nM T31721 CK7UW9 155519942 IC50 > 300000 nM T31721 C0Y9UF 155520160 IC50 > 300000 nM T31721 C52DFC 155524441 IC50 > 300000 nM T31721 C4IWE9 155525454 IC50 > 300000 nM T31721 CHJ5G1 155527881 IC50 > 300000 nM T31721 C9Z2ME 155529757 IC50 > 300000 nM T31721 CN1S4G 155530850 IC50 > 300000 nM T31721 C7HOI6 155533200 IC50 > 300000 nM T31721 CG65QS 155536541 IC50 > 300000 nM T31721 CX3ED4 155538143 IC50 > 300000 nM T31721 C4J3DC 155541203 IC50 > 300000 nM T31721 CD4B0V 155542542 IC50 > 300000 nM T31721 C87POT 155548017 IC50 > 300000 nM T31721 CPQM13 155555116 IC50 > 300000 nM T31721 CV9R4S 155557780 IC50 > 300000 nM T31721 C6NAQ5 155561202 IC50 > 300000 nM T31721 CF9YI6 155564787 IC50 > 300000 nM T31721 CFN45I 155565203 IC50 > 300000 nM T31721 CCK6T7 155565355 IC50 > 300000 nM T31721 CH9Q4R 44587874 IC50 = 2460 nM T31721 CRV3B2 44587876 IC50 = 21100 nM T31721 D02JJX 11531745 IC50 = 1862.09 nM T31721 D03RGP 1221 IC50 > 1000000 nM T31721 D03UIR 24905704 Ki = 3000 nM T31721 D04XZP 107883 IC50 > 3000000 nM T31721 D07GUB 5311218 IC50 = 7000 nM T31721 D09HET 11622683 IC50 = 10964.78 nM T31721 D0B2VW 95883 Ki = 5370.32 nM T31721 D0F5SO 11369932 IC50 = 420 nM T31721 D0JT2N 443239 IC50 = 9549.93 nM T31721 D0OT9B 5960 IC50 = 19498.45 nM T31721 D0X3CF 442879 IC50 > 500000 nM T13176 D03HUX 49792852 IC50 > 10000 nM T13176 D0H9FR 118295624 IC50 = 792 nM T13176 D0O0LS 25141092 IC50 > 10000 nM T13176 D0RX8U 86281829 IC50 = 0.7943 nM T13176 CD8J9V 11963346 IC50 = 42 nM T13176 CS3EB6 16044861 IC50 = 37.9 nM T13176 C0Z6VU 16045086 IC50 = 4.1 nM T13176 CA1T2U 16045087 IC50 = 820 nM T13176 C35ILP 16045759 IC50 = 9100 nM T13176 CQ4O0Y 16045761 IC50 = 142 nM T13176 C1VS7Q 16045839 IC50 = 54 nM T13176 CCFT24 16046014 IC50 = 86.7 nM T13176 C6QT0J 44622837 IC50 > 1000 nM T13176 CU3RF1 45139989 IC50 > 10000 nM T13176 CQGZ06 45139991 IC50 > 10000 nM T13176 C7ON5A 46233287 IC50 > 10000 nM T13176 CF91RS 49843531 IC50 > 10000 nM T13176 CY48DE 49849970 IC50 = 31 nM T13176 C2Y6QS 50938552 IC50 > 10000 nM T13176 C36LQJ 50940491 IC50 = 1100 nM T13176 CWN54R 51003389 IC50 = 250 nM T13176 C9NYP4 51036677 IC50 > 10000 nM T13176 C4WRY3 51037112 IC50 > 10000 nM T13176 CRI28Z 51037948 IC50 > 10000 nM T13176 C3LTA4 53317522 IC50 = 6800 nM T13176 C87OAQ 53317986 IC50 = 140 nM T13176 CM0N2P 53319337 IC50 = 1300 nM T13176 C1L8WR 53319339 IC50 = 840 nM T13176 CC2IW7 53320600 IC50 = 1300 nM T13176 CN1TI4 53320630 IC50 = 7800 nM T13176 CZN0B8 53320631 IC50 = 300 nM T13176 C92UFO 53321929 IC50 = 102 nM T13176 CY0V2M 53323287 IC50 = 2500 nM T13176 C4HKE1 53323288 IC50 = 1600 nM T13176 CA4T3Y 53323289 IC50 = 4200 nM T13176 CNW02P 53323290 IC50 = 350 nM T13176 CP41WD 53324073 IC50 = 823 nM T13176 CJ4G3Y 53324074 IC50 = 3500 nM T13176 CL4G1V 53324616 IC50 = 5000 nM T13176 CNO54Z 53324617 IC50 = 442 nM T13176 C1EXW0 53325922 IC50 = 16 nM T13176 C2JB0Z 53325923 IC50 = 556 nM T13176 CD03BA 53466725 IC50 = 5.4 nM T13176 CXB94H 53466728 IC50 = 11.7 nM T13176 CYQ41S 53466951 IC50 = 1.3 nM T13176 C7QJ9O 53467174 IC50 = 1.9 nM T13176 CK7HG1 53467177 IC50 = 0.6 nM T13176 C5LS6O 53467178 IC50 = 0.2 nM T13176 CDU2A9 53467392 IC50 = 0.9 nM T13176 C3EYH5 53467617 IC50 = 2.5 nM T13176 CEU1I5 53467819 IC50 = 1.2 nM T13176 C1RMJ9 53467824 IC50 = 0.7 nM T13176 C09RAS 53468037 IC50 = 0.5 nM T13176 C37YIA 53468254 IC50 = 0.4 nM T13176 CYXW95 53468661 IC50 = 1.9 nM T13176 CCBA89 53468860 IC50 = 100 nM T13176 CX0R1K 53469059 IC50 = 30 nM T13176 CV7C0D 53469060 IC50 < 30 nM T13176 CCKD45 53469061 IC50 = 2.7 nM T13176 C91STB 53469449 IC50 = 0.2 nM T13176 CV6P9J 53469453 IC50 = 0.2 nM T13176 C8FS3Q 53469629 IC50 = 0.2 nM T13176 C56MKE 53469634 IC50 = 0.9 nM T13176 CZ1CI3 53469824 IC50 = 100 nM T13176 C7R2AX 66561010 IC50 = 7.4 nM T13176 CD52SV 66561011 IC50 = 8.1 nM T13176 C6SEL2 66561012 IC50 = 1.5 nM T13176 CCJ25F 66561013 IC50 = 17.4 nM T13176 C9Q0PT 66561090 IC50 = 0.2 nM T13176 CIXK72 66561167 IC50 = 0.3 nM T13176 CJD4Z1 66823478 IC50 = 0.5 nM T13176 CKOE90 71451677 IC50 = 11 nM T13176 CCN01X 71547862 IC50 > 10000 nM T13176 CW2YU7 72704111 IC50 = 19.1 nM T13176 CWCA98 72704112 IC50 = 23.4 nM T13176 CPIH57 72704113 IC50 = 63.8 nM T13176 CH1X8Y 72704114 IC50 = 57.5 nM T13176 CV39OD 72704115 IC50 = 16.6 nM T13176 CH63PM 86281830 IC50 = 12.59 nM T13176 CJ9U3A 86281960 IC50 = 3.162 nM T13176 CX4H6I 86583042 IC50 = 41 nM T13176 CVR43W 86583044 IC50 = 9 nM T13176 CA81UY 86583045 IC50 = 84 nM T13176 CY0UC4 90645194 IC50 > 10000 nM T13176 C8GWQ4 117636459 IC50 = 251.19 nM T13176 CKA4U9 117636465 IC50 = 10 nM T13176 C9IN8R 117636472 IC50 = 0.3981 nM T13176 CI5L3E 117636490 IC50 = 6.31 nM T13176 C7M9VF 117636502 IC50 = 1.585 nM T13176 CH9E1Q 117636508 IC50 = 5.012 nM T13176 CY7BI2 118706214 IC50 > 10000 nM T13176 CC6T5H 118720605 IC50 = 0.631 nM T13176 C5QC8E 118730408 IC50 = 1 nM T13176 C4TXF2 118730409 EC50 = 520 nM T13176 CN2A9O 118730410 IC50 = 3 nM T13176 COF69K 118730411 IC50 = 1 nM T13176 CEJ1S6 118730412 IC50 = 240 nM T13176 CQ0T5Z 118730413 IC50 = 140 nM T13176 CF47CO 118730414 EC50 = 130 nM T13176 CEJ67D 118730415 EC50 = 200 nM T13176 C5SI6Q 118730416 IC50 = 5 nM T13176 CR0H9D 118730417 IC50 = 240 nM T13176 CGDW48 118730418 EC50 = 190 nM T13176 C23KFD 118730419 IC50 = 11 nM T13176 CJ9SA8 118730420 IC50 = 53 nM T13176 C0HK5A 118730421 IC50 = 79 nM T13176 C1Q0UN 118730422 EC50 = 1300 nM T13176 C1K0PE 118730423 IC50 = 12 nM T13176 CHA4N2 136013680 IC50 > 10 nM T13176 C3COS8 136160805 IC50 = 18 nM T13176 C1YUD0 136219394 IC50 > 10 nM T13176 CIU8W3 136254389 IC50 > 10 nM T13176 C2MD1Q 155513187 IC50 > 10000 nM T13176 D08HFG 24809764 IC50 > 10000 nM T13176 D09HVH 135566652 IC50 > 10 nM T13176 D0N4LR 53469448 IC50 < 30 nM T59550 C13QNP 65127 IC50 = 11500 nM T59550 COEW50 439427 IC50 > 10000 nM T59550 CCK25W 10070969 IC50 = 46500 nM T59550 CL7R6H 10102934 IC50 = 90 nM T59550 C64LCF 44449242 IC50 = 20000 nM T59550 CJ9QO3 44449275 IC50 = 1800 nM T59550 CJY5X7 44449622 IC50 = 3700 nM T59550 C5P6RV 44449654 IC50 = 4440 nM T59550 C3NW7E 44449688 IC50 = 5030 nM T59550 C1X2JY 44449727 IC50 = 4760 nM T59550 CQ54JK 135410197 IC50 = 77100 nM T59550 CRT3X6 135524445 IC50 = 3200 nM T73859 CQTJ86 9547099 EC50 = 245.47 nM T73859 CIY57T 9547100 EC50 = 288.4 nM T73859 C6L2IH 44475675 EC50 = 1659.59 nM T73859 CE2FR8 52926276 EC50 = 831.76 nM T73859 CK6IV9 52926277 EC50 > 1000 nM T73859 CSV34F 52926278 EC50 = 1348.96 nM T73859 CJI7F3 71495077 EC50 > 1000 nM T73859 CW9DS0 78319779 EC50 = 150 nM T73859 CVM0N2 122177490 EC50 = 410 nM T73859 C5U2LP 122177491 EC50 > 1000 nM T73859 C02ODQ 122177492 EC50 = 316.23 nM T73859 C0PF6Z 122177493 EC50 > 1000 nM T73859 CQ4H8Y 122177494 EC50 > 1000 nM T73859 CC43DK 122177497 EC50 = 3100 nM T73859 C2BWT6 122177498 EC50 > 1000 nM T73859 C4C1RL 122177499 EC50 = 700 nM T73859 CC7DB0 122177500 EC50 > 1000 nM T73859 CH69GX 122177501 EC50 > 1000 nM T73859 C51KDV 122177502 EC50 > 1000 nM T73859 C5L3NY 122177503 EC50 > 1000 nM T73859 CEZN81 122177504 EC50 > 1000 nM T73859 C2TQ8R 122177513 EC50 > 1000 nM T73859 CAZ90F 122177516 EC50 = 930 nM T73859 C4JP1B 122177517 EC50 = 457.09 nM T73859 CLD62P 122177520 EC50 = 234.42 nM T73859 CA8ZJ5 122177521 EC50 = 158.49 nM T73859 C67LAE 122177522 EC50 > 1000 nM T73859 C30HEC 122177523 EC50 > 1000 nM T73859 CJ0RD5 122177524 EC50 = 1800 nM T73859 C6GI8E 122177525 EC50 > 1000 nM T73859 C0C5XU 122177526 EC50 > 1000 nM T73859 C74WRP 122177527 EC50 > 1000 nM T73859 C61RUZ 122177528 EC50 = 933.25 nM T73859 CRZ1V8 122177589 EC50 > 1000 nM T73859 CHM1G0 137633515 EC50 = 229.09 nM T73859 C32PCR 137640053 EC50 = 90 nM T73859 C7GJI8 137641921 EC50 = 295.12 nM T73859 CPVC58 137644526 EC50 = 77.62 nM T73859 C13SGK 137645387 EC50 = 180 nM T73859 CF0BR4 137652635 EC50 = 14.79 nM T73859 C8EKO2 137655293 EC50 = 26.92 nM T73859 C7UTX3 137660207 EC50 = 40.74 nM T74607 CEU84H 67070 IC50 = 18000 nM T74607 CGO87D 109515 IC50 = 1700 nM T74607 C31TOA 272513 IC50 = 400 nM T74607 CLO34W 345609 IC50 = 1900 nM T74607 CA4X9B 389769 IC50 = 7900 nM T74607 CDW4H7 919981 IC50 = 1200 nM T74607 C21FTE 2725176 IC50 = 600 nM T74607 CKT8H4 2735844 IC50 > 300000 nM T74607 CXG38R 6077765 IC50 = 4400 nM T74607 C75POE 10705175 IC50 = 1700 nM T74607 C4UH0J 11191273 IC50 = 400 nM T74607 CSZ95E 11736269 IC50 = 3800 nM T74607 CC30DG 12099906 IC50 = 1600 nM T74607 CCL89N 15712171 IC50 = 10700 nM T74607 CJ4Y1K 54293327 IC50 = 1800 nM T74607 CZ21OQ 70533134 IC50 = 13500 nM T74607 CW5Q0B 71561829 IC50 > 300000 nM T74607 C0AEW4 71561950 IC50 > 300000 nM T74607 CGD03K 71561951 IC50 = 700 nM T74607 CR49ZS 71561952 IC50 > 300000 nM T74607 CTS61D 71561953 IC50 > 300000 nM T74607 CN63ED 71561954 IC50 > 300000 nM T74607 C9E3FZ 71561955 IC50 > 300000 nM T74607 C25SAJ 71561956 IC50 > 300000 nM T74607 CMW82G 71562076 IC50 > 300000 nM T74607 CX2Z3E 71562077 IC50 = 900 nM T74607 CQK24E 71562078 IC50 = 400 nM T74607 CY5VZ9 71562079 IC50 = 500 nM T74607 CDM8W9 71562080 IC50 = 4000 nM T74607 CUBM18 71562081 IC50 = 8000 nM T74607 C3OR8G 71562082 IC50 = 8000 nM T74607 C3M9HF 71562083 IC50 > 300000 nM T74607 CDC7S6 71562084 IC50 = 5300 nM T74607 CWA7T5 71562200 IC50 = 4700 nM T74607 C6J0QL 71562201 IC50 = 1300 nM T74607 CE4P3O 71562202 IC50 > 300000 nM T74607 CYO16E 71562203 IC50 = 10800 nM T74607 CA2RE1 71562204 IC50 = 3800 nM T74607 CLB8Q7 71562205 IC50 = 8900 nM T74607 CL5XA2 71562310 IC50 = 12600 nM T74607 C3WFG6 71562311 IC50 = 2400 nM T74607 CLT3N5 71712196 IC50 = 4000 nM T74607 C6AV3D 73669655 IC50 = 17000 nM T74607 CGRX70 73669656 IC50 = 17100 nM T74607 C0K8PF 117027088 IC50 = 34000 nM T74607 CG23HU 124203912 IC50 = 400 nM T74607 CLY73N 127043180 IC50 = 2200 nM T74607 COKC35 127043186 IC50 = 2900 nM T74607 CJ3B7A 127043193 IC50 = 500 nM T74607 CR94NM 127043560 IC50 = 5700 nM T74607 CO07LC 127044218 IC50 = 8700 nM T74607 CD9BN8 127044543 IC50 = 3600 nM T74607 CE60FV 127044544 IC50 = 1400 nM T74607 CYK2G6 127044578 IC50 = 700 nM T74607 CC2TQ1 127044703 IC50 = 5800 nM T74607 CTBN78 127044709 IC50 = 1500 nM T74607 C3HTN2 127044710 IC50 = 1100 nM T74607 C7GLS6 127044711 IC50 = 2700 nM T74607 CHK70L 127044712 IC50 = 1000 nM T74607 CKA4S7 127044759 IC50 = 2900 nM T74607 CMO07X 127044874 IC50 = 1300 nM T74607 CWO7V8 127044876 IC50 = 1100 nM T74607 C8PWJ6 127045030 IC50 = 3300 nM T74607 C2BL8R 127045043 IC50 = 1800 nM T74607 CY4OJ8 127045044 IC50 = 1800 nM T74607 CM94PU 127045045 IC50 = 2000 nM T74607 C1J3FD 127045046 IC50 > 300000 nM T74607 CYWZ03 127045181 IC50 = 3000 nM T74607 CSF5C0 127045202 IC50 = 46000 nM T74607 CZDL62 127045412 IC50 = 1800 nM T74607 CL28CD 135348458 IC50 = 2500 nM T74607 C1C9RT 135348459 IC50 = 2500 nM T74607 CKL53Z 135348461 IC50 = 28400 nM T74607 CW4GV0 135348495 IC50 = 6300 nM T74607 CIJX92 135348498 IC50 = 3400 nM T74607 C8HRN2 135348503 IC50 = 12400 nM T74607 CUT6Q0 135348509 IC50 = 15800 nM T74607 C7G8IC 135348516 IC50 = 5400 nM T74607 CT2HM9 135348563 IC50 = 3000 nM T74607 CKXT68 135348703 IC50 = 1200 nM T74607 CT01FH 135434170 IC50 = 30500 nM T74607 CDY4R5 135473051 IC50 = 8400 nM T74607 CRHL91 136226115 IC50 > 300000 nM T74607 CHI5S6 136226117 IC50 = 12700 nM T74607 CYC91X 136226118 IC50 = 15700 nM T74607 CC7DG5 136226119 IC50 > 300000 nM T74607 C3DQW5 136226120 IC50 = 11600 nM T74607 CX4J2V 136226121 IC50 = 127000 nM T74607 CZ0AR1 136226122 IC50 > 300000 nM T74607 C8GLQ1 136228202 IC50 = 7000 nM T74607 C9RC1Q 136228203 IC50 = 4000 nM T74607 CBYW70 136228204 IC50 = 5900 nM T74607 C94MYO 136244206 IC50 = 38700 nM T74607 C32ZQT 136244263 IC50 > 300000 nM T74607 CQ4N5W 136244264 IC50 > 300000 nM T74607 C4QA8F 136254218 IC50 > 300000 nM T74607 CB90NH 136254219 IC50 > 300000 nM T74607 D00EHP 22200891 IC50 = 300 nM T74607 D0GP7D 54686376 IC50 = 3800 nM T74607 D0UB2J 6076 IC50 = 40000 nM T66665 D00IBN 54676228 IC50 = 218000 nM T66665 D03RTS 2662 IC50 = 0.52 nM T66665 D04AIT 5280445 IC50 = 2.5 ug.mL-1 T66665 D04YMH 151166 IC50 = 7 nM T66665 D05FTJ 4044 IC50 = 2900 nM T66665 D05UWI 119828 IC50 = 5 nM T66665 D05VLS 5090 IC50 = 1 nM T66665 D06YPU 39912 IC50 = 730 nM T66665 D07BPS 5359 IC50 = 2750 nM T66665 D07POC 176870 IC50 > 10000 nM T66665 D08IFL 4037 IC50 = 40 nM T66665 D09JUG 60490 IC50 > 10000 nM T66665 D09MGR 123619 IC50 = 81 nM T66665 D0A1PX 3394 IC50 = 10 nM T66665 D0B2WJ 3371 IC50 = 9300 nM T66665 D0C4YC 4075 IC50 = 7530 nM T66665 D0D9JW 3826 IC50 = 140 nM T66665 D0DJ1B 156391 IC50 = 900 nM T66665 D0G7FJ 54677470 IC50 = 700 nM T66665 D0GY5Z 2244 IC50 = 2400 nM T66665 D0I0EG 44093 Ki = 12000 nM T66665 D0IT2X 2581 IC50 = 100 nM T66665 D0K8KX 5280343 IC50 = 28600 nM T66665 D0L6DA 119607 IC50 = 5 nM T66665 D0M9DC 4614 IC50 = 110 nM T66665 D0N1WU 3308 IC50 = 2000 nM T66665 D0R1QE 3672 IC50 = 1100 nM T66665 D0R1RS 3715 IC50 = 5.9 nM T66665 D0TG1H 3033 IC50 = 5 nM T66665 D0U5QK 1983 IC50 = 141000 nM T66665 D0W9WF 3825 IC50 = 26 nM T66665 D0Z5IU 1548887 IC50 = 8800 nM T66665 D02DYU 9858913 IC50 = 62 nM T66665 D05FGR 92337 IC50 = 123000 nM T66665 D0C5DC 72099 IC50 = 910 nM T66665 D0I6LH 107985 IC50 = 40 nM T66665 D0LI1C 44469321 IC50 > 30000 nM T66665 D0U3EP 445154 IC50 = 990 nM T66665 D0U8OD 213053 IC50 = 66 nM T66665 D0DK4I 4534 IC50 > 50000 nM T66665 D0KG9M 19910 Ki = 1000 nM T66665 D0M6LX 56851703 IC50 > 100000 nM T66665 D0O4QB 3314 IC50 = 129000 nM T66665 D00RSK 9832687 IC50 = 3 nM T66665 D02OHR 443373 IC50 = 25.7 nM T66665 D03NZV 9865808 IC50 = 10 nM T66665 D05EYG 9799453 IC50 = 140 nM T66665 D05MCS 44473151 IC50 > 100000 nM T66665 D05REH 71246 IC50 = 21 nM T66665 D05WPQ 6438354 IC50 > 10 nM T66665 D07HBI 132306 IC50 > 100000 nM T66665 D07TZM 115239 IC50 = 90 nM T66665 D08GRY 3177 IC50 = 2 nM T66665 D09BKE 4553 IC50 = 1 nM T66665 D0C0JT 4495 IC50 = 15 nM T66665 D0K2ER 3651377 IC50 > 10 nM T66665 D0N1SU 133021 IC50 = 370 nM T66665 D0O9JX 9851770 IC50 = 7.5 nM T66665 D0P3KA 60542 IC50 = 100 nM T66665 D0Z5LZ 159271 IC50 = 85 nM T66665 CUJY61 9948196 IC50 = 4930 nM T66665 CZB0X2 44411662 IC50 = 4220 nM T66665 CPU3K6 16007230 IC50 = 920 nM T66665 C7L5FX 44413160 IC50 = 2100 nM T66665 C0U5TZ 1302 IC50 = 280 nM T66665 C21TXQ 2151 IC50 = 42000 nM T66665 C1S7VI 2415 IC50 > 33000 nM T66665 C8IB3S 3965 IC50 = 13500 nM T66665 CU1X7Z 4237 IC50 = 440 nM T66665 CB4CP6 7115 IC50 = 144000 nM T66665 C9KD6A 10189 IC50 = 20100 nM T66665 CV24FH 10228 IC50 = 81100 nM T66665 CCF85O 10774 IC50 = 10000 nM T66665 CQP80E 15339 IC50 = 250 nM T66665 CGU07V 22633 IC50 = 700 nM T66665 C8YOP9 22810 IC50 = 21 nM T66665 C4EJ7D 27022 IC50 > 10000 nM T66665 CRVG43 27023 IC50 = 330 nM T66665 CKX05O 27861 IC50 = 100 nM T66665 CTY1P6 28566 IC50 = 530 nM T66665 CS51BE 31164 IC50 = 17200 nM T66665 CMZ01B 37486 IC50 = 340 nM T66665 CVS6A8 40634 IC50 = 150 nM T66665 CA1H6W 50204 IC50 = 50 nM T66665 CME3K9 65048 IC50 > 40000 nM T66665 CPW9B5 65752 IC50 = 300 nM T66665 CYI58D 72185 IC50 = 2300 nM T66665 C7IA0L 72540 IC50 = 400 nM T66665 CQT19P 73641 IC50 > 40000 nM T66665 C7VSL6 76743 IC50 = 4000 nM T66665 CGF95Y 78363 IC50 > 100000 nM T66665 C6NLX4 84003 IC50 = 120 nM T66665 CHJK85 85393 IC50 = 130 nM T66665 CZ8U6A 87020 IC50 > 100000 nM T66665 CA3RJ2 95686 IC50 = 2000 nM T66665 C2IRA6 127923 IC50 = 480 nM T66665 C1YCW7 129439 IC50 = 200 nM T66665 C6JI9T 151610 IC50 = 400 nM T66665 CF2O4N 158143 IC50 > 10000 nM T66665 CPS7E0 159665 IC50 = 5000 nM T66665 CW8K1N 168928 IC50 > 40000 nM T66665 C6A0PT 169118 IC50 > 25000 nM T66665 CDC52U 169187 IC50 > 50000 nM T66665 C2KD9Z 171596 IC50 > 50000 nM T66665 C02HKG 177140 IC50 = 3800 nM T66665 C6L5AP 181271 IC50 > 40900 nM T66665 CC2W4T 182489 IC50 = 90 nM T66665 CYWS98 185848 IC50 = 22300 nM T66665 CX41GY 189866 IC50 = 1000 nM T66665 CGUW53 196841 IC50 = 65000 nM T66665 CYTV54 227830 IC50 = 18000 nM T66665 C2W3TD 263547 IC50 = 180 nM T66665 CJ0MV1 291096 IC50 = 2900 nM T66665 C93TLF 297850 IC50 = 1000 nM T66665 C6AKQ8 308411 IC50 = 3360 nM T66665 CM2B0E 377558 IC50 = 5000 nM T66665 C8HA5W 404196 IC50 = 12420 nM T66665 CQCK56 404197 IC50 = 16850 nM T66665 C8BCZ1 404198 IC50 = 2040 nM T66665 CC20HA 404319 IC50 = 2930 nM T66665 C1MKV8 404320 IC50 = 3400 nM T66665 CI1GD8 404323 IC50 = 3090 nM T66665 COU8H0 404325 IC50 = 4600 nM T66665 C56XBC 404376 IC50 = 2730 nM T66665 CFJX25 405488 IC50 = 4280 nM T66665 CJTR17 405491 IC50 = 740 nM T66665 C01ANL 405559 IC50 = 2850 nM T66665 C3PZ1R 405561 IC50 = 2950 nM T66665 C9K5UB 441677 IC50 > 10000 nM T66665 CB60GF 442700 IC50 > 46700 nM T66665 CEI08Y 443378 IC50 = 34 nM T66665 C65MQP 443639 IC50 = 69700 nM T66665 C26UHG 470258 IC50 = 250000 nM T66665 CZ30UN 471843 IC50 > 40000 nM T66665 CB56XC 480869 IC50 > 100000 nM T66665 C7I8NK 484757 IC50 = 80000 nM T66665 CPJ59X 572426 IC50 > 100000 nM T66665 CCI7B9 572427 IC50 > 100000 nM T66665 CZ7O3I 636928 IC50 = 9500 nM T66665 CA9BW2 637234 IC50 > 40000 nM T66665 C5YS3J 637775 IC50 = 28000 nM T66665 CQ94TR 639465 IC50 = 4200 nM T66665 CMJ91Y 667550 IC50 = 27 nM T66665 C9H8UF 667685 IC50 = 5300 nM T66665 CO5W9I 684847 IC50 = 410 nM T66665 CLH9V1 690276 IC50 = 1390 nM T66665 CATJ47 722563 IC50 > 5000 nM T66665 C28PTM 724576 IC50 = 3690 nM T66665 CZN6S9 743974 IC50 > 100000 nM T66665 C96AHO 768025 IC50 = 1370 nM T66665 CPM12N 775994 IC50 > 100000 nM T66665 CC9K1G 779202 IC50 = 1200 nM T66665 CW14ZC 827480 IC50 > 100000 nM T66665 CO7NG6 867556 IC50 > 5000 nM T66665 C1V7BH 871573 IC50 = 130.4 nM T66665 C19IVK 873121 IC50 > 5000 nM T66665 C7U3CX 873133 IC50 = 840 nM T66665 CU0Y2L 914352 IC50 = 30400 nM T66665 C60RDY 973003 IC50 = 1080 nM T66665 C31WJN 1110835 IC50 = 1340 nM T66665 CILN42 1356792 IC50 > 10000 nM T66665 CYTU15 1370268 IC50 = 460 nM T66665 CMYK57 1500232 IC50 = 18200 nM T66665 C84MXV 1500233 IC50 = 15800 nM T66665 CWNY21 1500235 IC50 = 8000 nM T66665 C32RIC 1506603 IC50 = 60 nM T66665 CI26ZE 1514885 IC50 = 1500 nM T66665 CADY74 1517275 IC50 > 100000 nM T66665 C9B3KF 1850249 IC50 = 440 nM T66665 C31ILB 1856731 IC50 = 270 nM T66665 C1PHK6 2058278 EC50 = 330 nM T66665 CD89GA 2083607 IC50 = 2400 nM T66665 C10XPM 2127532 IC50 = 63 nM T66665 CO85TF 2254772 IC50 > 5000 nM T66665 C1K2QE 2317371 IC50 > 100000 nM T66665 C21JKB 2331369 IC50 = 56 nM T66665 CJDQ70 2731332 IC50 = 390 nM T66665 CN9AS5 2756535 IC50 > 100000 nM T66665 CT6W1B 2765724 IC50 = 60.26 nM T66665 CQUB26 2801736 IC50 > 300000 nM T66665 C9LOJ7 2826057 IC50 = 1120 nM T66665 CL5N8W 2896983 IC50 = 40 nM T66665 CQM64G 3037018 IC50 = 5500 nM T66665 CX6D4S 3058754 IC50 = 50 nM T66665 CXA70K 3080594 IC50 = 138000 nM T66665 CP4IL0 3629561 IC50 = 11340 nM T66665 C1M3TK 3954928 IC50 = 350 nM T66665 CL9BO3 4090966 IC50 = 120 nM T66665 CY2XM7 4226790 IC50 = 330 nM T66665 C23MOL 4308557 IC50 = 4000 nM T66665 C5LQ3D 4322149 IC50 > 20000 nM T66665 CM9H6J 4434869 IC50 = 52 nM T66665 C8GF1S 4460526 IC50 = 18500 nM T66665 CSEJ76 4521790 IC50 = 810 nM T66665 CA9X7C 4679898 IC50 = 150 nM T66665 CAKX74 4763851 IC50 = 740 nM T66665 C4JQ5B 4763963 IC50 > 100000 nM T66665 CJ74EB 4990103 IC50 = 3500 nM T66665 CNPV35 5018304 IC50 = 800 nM T66665 CVT05I 5080393 IC50 > 100000 nM T66665 C0IS9Y 5100138 IC50 = 120.23 nM T66665 CDU89L 5195985 IC50 = 151.4 nM T66665 C1DR8C 5281479 IC50 = 1100 nM T66665 C0D3PO 5281671 IC50 = 100000 nM T66665 CMAH08 5315472 IC50 = 36370 nM T66665 CRL9M3 5319925 IC50 = 2500 nM T66665 CNX87V 5320767 IC50 = 4600 nM T66665 CJ8P4T 5352624 IC50 = 100 nM T66665 CJC3M8 5378591 IC50 = 7522 nM T66665 CSOV90 5386591 IC50 = 3400 nM T66665 CH6DT9 5481958 IC50 > 100000 nM T66665 CWS5X0 5481970 IC50 > 100000 nM T66665 C7B1CG 5487413 IC50 = 8000 nM T66665 C8M0OD 5716903 IC50 = 6000 nM T66665 CUYR71 6050842 IC50 = 4017 nM T66665 CS03BA 6255462 IC50 = 19600 nM T66665 C9J6LF 6426663 IC50 = 32 nM T66665 C0GZU8 6426686 IC50 = 300 nM T66665 CF8E2M 6444394 IC50 = 4700 nM T66665 CZ49FU 6997572 IC50 > 100000 nM T66665 CH7GX6 7005167 IC50 = 55000 nM T66665 CXQ86B 7019898 IC50 = 80 nM T66665 C4K3IT 7732606 IC50 = 130 nM T66665 CRF4L8 7732607 IC50 = 110 nM T66665 CS5Y9N 7964055 IC50 > 17000 nM T66665 CC97TP 7972918 IC50 = 260 nM T66665 C3BU5H 8566717 IC50 > 100000 nM T66665 C5TH6L 8778611 IC50 = 25000 nM T66665 CLF8W5 9559931 IC50 = 802320 nM T66665 CB7LR9 9644405 IC50 = 203690 nM T66665 C0NTV6 9795652 IC50 = 320 nM T66665 CC38MG 9796843 IC50 = 170 nM T66665 C9MX1U 9797752 IC50 = 2197.86 nM T66665 C08TVM 9797804 IC50 = 0.12 nM T66665 C24SGI 9798392 IC50 = 15 nM T66665 CSQD86 9799387 IC50 = 436.52 nM T66665 C1N8HK 9800211 IC50 = 10 nM T66665 C2XRG4 9800221 IC50 = 1200 nM T66665 CSA4F1 9800270 IC50 = 10 nM T66665 C64NBT 9801204 IC50 = 7.943 nM T66665 CV5S6A 9801701 IC50 < 6 nM T66665 CXEU61 9802596 IC50 = 365 nM T66665 C4FY8C 9803430 IC50 = 190 nM T66665 C59KTP 9803459 IC50 = 235 nM T66665 CZQ60H 9813036 IC50 = 200000 nM T66665 CXA90U 9813147 IC50 = 66000 nM T66665 CZ8FD1 9813916 IC50 = 11000 nM T66665 CZT7M2 9816662 IC50 = 10 nM T66665 CC6A2L 9817667 IC50 = 1.2 nM T66665 CV5Y2H 9818233 IC50 = 11 nM T66665 C2AKX0 9818254 IC50 = 300000 nM T66665 CQK3E5 9818359 IC50 = 2398.83 nM T66665 C46ENF 9818598 IC50 = 5200 nM T66665 C03FBZ 9818888 IC50 = 180 nM T66665 CZ0K8H 9819804 IC50 = 80 nM T66665 C9RST2 9821264 IC50 = 14 nM T66665 CW37TE 9821646 IC50 = 109.65 nM T66665 CNC0P9 9822123 IC50 = 1234809.61 nM T66665 CUO02B 9822332 IC50 = 60.26 nM T66665 CC75ZO 9822357 IC50 = 18 nM T66665 C3ZTC7 9822818 IC50 = 4.677 nM T66665 CS96DK 9822874 IC50 = 30 nM T66665 CE4Y8C 9822883 IC50 = 728 nM T66665 CB0Y6K 9823368 IC50 = 1730 nM T66665 CV7T4Q 9823594 IC50 = 6 nM T66665 CEH01K 9823932 IC50 = 4000 nM T66665 CIZ04N 9825026 IC50 = 700 nM T66665 C7MYZ9 9825432 IC50 = 8.913 nM T66665 C20MHW 9825527 IC50 = 60 nM T66665 C8FW0R 9825900 IC50 = 40 nM T66665 CP94CU 9831791 IC50 = 10 nM T66665 C4FS6L 9834940 IC50 = 250000 nM T66665 CE8A4O 9835301 IC50 = 7000 nM T66665 CEGR47 9835721 IC50 = 51 nM T66665 CUT4N2 9836619 IC50 = 7 nM T66665 CISH24 9836698 IC50 = 30 nM T66665 CZG4J5 9838569 IC50 = 230 nM T66665 CHNX31 9839177 IC50 = 45000 nM T66665 C2TPB6 9839884 IC50 = 12000 nM T66665 CD9YC2 9840237 IC50 = 300 nM T66665 C1BXD4 9840568 IC50 = 100 nM T66665 CK65IB 9840638 IC50 = 6500 nM T66665 C23HSC 9841079 IC50 = 15 nM T66665 C2NDG3 9841276 IC50 = 130 nM T66665 CA1YN6 9841715 IC50 = 1069.05 nM T66665 CA9IV0 9842523 IC50 = 21.5 nM T66665 C8Y4ND 9842547 IC50 = 2147.83 nM T66665 C6U5CF 9842936 IC50 = 2818.38 nM T66665 C6HDX1 9842937 IC50 = 510 nM T66665 CF15GO 9843089 IC50 = 40.74 nM T66665 CJIN69 9843189 IC50 > 10000 nM T66665 C4RSA3 9843356 IC50 = 1.995 nM T66665 CA1TD9 9843737 IC50 = 3450 nM T66665 CMX5B4 9844547 IC50 = 130 nM T66665 C34IOV 9846219 IC50 = 4700 nM T66665 C94NVU 9846581 IC50 = 20 nM T66665 C5A6OB 9847751 IC50 = 60 nM T66665 CCV9U2 9849164 IC50 = 500 nM T66665 CTMX24 9857378 IC50 = 50000 nM T66665 CXQ6E3 9858164 IC50 = 620 nM T66665 CP75VI 9861581 IC50 = 12000 nM T66665 CS6Y5U 9861661 IC50 = 220 nM T66665 CJLR90 9861712 IC50 > 10000 nM T66665 C5AP3Q 9861854 IC50 = 70 nM T66665 CV57DI 9861888 IC50 = 70 nM T66665 CX87MB 9863426 IC50 = 2180 nM T66665 C5NG2Y 9863475 IC50 = 10000000 nM T66665 C49BAD 9864100 IC50 = 19.2 nM T66665 C2TP7H 9865298 IC50 = 80 nM T66665 CP4QG9 9865547 IC50 = 7.943 nM T66665 C27YKN 9865599 IC50 = 1000 nM T66665 C5CW2O 9867708 IC50 = 570 nM T66665 C7ZEH1 9868819 IC50 = 2500 nM T66665 CMNZ15 9869703 IC50 = 120 nM T66665 CA43PC 9871042 IC50 = 50 nM T66665 C8PHY4 9871438 IC50 > 1000 nM T66665 CSE53Z 9878306 IC50 = 31600 nM T66665 CY1AR6 9880758 IC50 = 48.98 nM T66665 CUW93O 9883082 IC50 = 11000 nM T66665 CP2NZ0 9883585 IC50 = 0.08 nM T66665 C43HGV 9883653 IC50 = 140 nM T66665 C1FOR4 9883749 IC50 > 10000 nM T66665 CS6HN1 9883822 IC50 = 2.8 nM T66665 C8U7TB 9883880 IC50 = 29 nM T66665 C29QLY 9884031 IC50 = 47 nM T66665 CYU2N6 9884096 IC50 = 1499.68 nM T66665 CZF0A2 9884371 IC50 = 100 nM T66665 CMV92I 9885354 IC50 = 12.88 nM T66665 C9IZG0 9888058 IC50 = 150 nM T66665 CFV10P 9889157 IC50 = 4000 nM T66665 C87ODI 9890350 IC50 = 75.86 nM T66665 C4UBC3 9891184 IC50 = 650 nM T66665 CP8C5S 9899321 IC50 = 20000 nM T66665 CGIN75 9899360 IC50 = 34000 nM T66665 C78JRI 9899469 IC50 = 5000 nM T66665 C59BYV 9899638 IC50 > 40000 nM T66665 CEB3O9 9900153 IC50 = 100000 nM T66665 CV0SP3 9901158 IC50 = 120 nM T66665 CILP75 9901319 IC50 = 41 nM T66665 CU21FI 9902732 IC50 = 101 nM T66665 C9ON6P 9902810 IC50 = 120.23 nM T66665 CQL3O0 9903494 IC50 = 7000 nM T66665 C7JE5S 9904089 IC50 > 10000 nM T66665 C2SRN6 9905412 IC50 = 263.03 nM T66665 COA31Z 9905676 IC50 = 510.5 nM T66665 CB1D4T 9905741 IC50 = 5 nM T66665 C2YDI0 9905875 IC50 = 400 nM T66665 CZ30RH 9906073 IC50 = 3700 nM T66665 CAH7V1 9906472 IC50 = 10 nM T66665 CT4JM6 9907429 IC50 = 700 nM T66665 C4P5DV 9907758 IC50 = 27 nM T66665 CG8P5T 9908624 IC50 = 10 nM T66665 C2T6IY 9908677 IC50 = 860 nM T66665 C7L2XS 9908988 IC50 = 250 nM T66665 C1SEB7 9909016 IC50 = 470 nM T66665 CQ83VI 9909642 IC50 < 21 nM T66665 CVUP23 9910697 IC50 = 50 nM T66665 CW2S5L 9911248 IC50 = 400 nM T66665 CS4YT5 9912793 IC50 = 200 nM T66665 CC2J3T 9918019 IC50 = 1000 nM T66665 CD0J1F 9918457 IC50 = 19 nM T66665 CH8LW6 9921698 IC50 = 7000 nM T66665 C05YIR 9921835 IC50 = 50000 nM T66665 C0Y5BR 9922118 IC50 = 190 nM T66665 CE2LZ0 9922659 IC50 = 240 nM T66665 CWJH86 9922739 IC50 = 3200 nM T66665 CZ0IQ2 9923656 IC50 = 1800 nM T66665 CSU35P 9924251 IC50 = 218.78 nM T66665 C06GJS 9925288 IC50 = 40 nM T66665 C5C9DS 9925578 IC50 = 470 nM T66665 C42GTD 9926659 IC50 = 39000 nM T66665 C8TA9U 9926877 IC50 = 320 nM T66665 CR8TW5 9927594 IC50 = 3 nM T66665 C2QSC1 9927613 IC50 = 30 nM T66665 CK71LW 9927909 IC50 = 1840 nM T66665 CG1C3L 9927912 IC50 = 2.6 nM T66665 CY1F3R 9928047 IC50 = 3 nM T66665 CXY6V4 9928340 IC50 = 319.89 nM T66665 C2OUH1 9928381 IC50 = 1199.5 nM T66665 C70GRD 9928539 IC50 = 16 nM T66665 COE0X2 9928728 IC50 = 3369.77 nM T66665 C2CJ4G 9929140 IC50 = 1690 nM T66665 C8Z3SJ 9929308 IC50 = 13 nM T66665 CS7EB8 9929562 IC50 = 50 nM T66665 CT0HB7 9929697 IC50 = 15 nM T66665 C8N4FQ 9930747 IC50 = 1700 nM T66665 CHS01T 9930803 IC50 = 0.5 nM T66665 C9HQ1Z 9931215 IC50 = 0.25 nM T66665 CAOW72 9931274 IC50 = 6919.9 nM T66665 CUVI39 9932045 IC50 = 6 nM T66665 CS2ZH4 9932828 IC50 = 30 nM T66665 C6QPN2 9933112 IC50 = 50 nM T66665 CJ4AV0 9933456 IC50 = 52 nM T66665 CBE54A 9934809 IC50 = 220 nM T66665 CY1C2F 9935923 IC50 = 58 nM T66665 C97YOJ 9936231 IC50 = 50 nM T66665 CY7V9W 9937470 IC50 = 0.3 nM T66665 CWJ05V 9942490 IC50 = 25000 nM T66665 C6RQW1 9945282 IC50 = 39000 nM T66665 CU6J7M 9945403 IC50 = 75 nM T66665 CXK27R 9946200 IC50 = 239.88 nM T66665 CF9QL0 9946917 IC50 = 120 nM T66665 CH7ZK2 9947111 IC50 = 141.25 nM T66665 CWU4Y1 9947165 IC50 = 830 nM T66665 CQC75N 9947305 IC50 = 120 nM T66665 CYQF10 9947309 IC50 = 870 nM T66665 CIC92Y 9947371 IC50 = 1500 nM T66665 CKWB53 9947925 IC50 = 950 nM T66665 CITM37 9947934 IC50 = 60 nM T66665 C4WC8T 9948569 IC50 = 620 nM T66665 C42BFH 9949984 IC50 = 690 nM T66665 C0GC2F 9950666 IC50 = 1530 nM T66665 C87QWC 9950669 IC50 = 20 nM T66665 CUV05Z 9954100 IC50 = 75 nM T66665 CL1W0Y 9954883 IC50 = 100 nM T66665 C1IN3C 9955928 IC50 = 150 nM T66665 C0RTJ9 9956213 IC50 = 55 nM T66665 C1KJ3G 9956925 IC50 = 40 nM T66665 CAU01B 9957131 IC50 = 45 nM T66665 C04ZJC 9965352 IC50 = 100000 nM T66665 CZN2B4 9966560 IC50 = 62 nM T66665 CMF25N 9967049 IC50 = 350 nM T66665 CO5Y8D 9967335 IC50 = 12000 nM T66665 C25VMC 9967345 IC50 = 70 nM T66665 CQX38P 9967467 IC50 = 5500 nM T66665 CS8VF5 9967867 IC50 = 338.84 nM T66665 CA8E7F 9968075 IC50 = 2300 nM T66665 CIPL92 9968334 IC50 > 40000 nM T66665 CP5O2E 9969153 IC50 = 10000 nM T66665 C5XM8F 9969968 IC50 = 400 nM T66665 C4K0IL 9970134 IC50 = 1540 nM T66665 C4AUM2 9973893 IC50 = 8700 nM T66665 CF50NP 9982906 IC50 = 55670 nM T66665 CDA38U 9987332 IC50 = 73000 nM T66665 CO68GP 9993267 IC50 = 300 nM T66665 CQO56T 9993978 IC50 > 100000 nM T66665 CJ9E2P 9998267 IC50 = 500 nM T66665 COQ5S1 10000662 IC50 = 92300 nM T66665 CWY7U3 10001441 IC50 = 350 nM T66665 C6FM2Z 10001804 IC50 = 20 nM T66665 CPR56D 10005148 IC50 = 1513.56 nM T66665 CMJH05 10016051 IC50 = 730 nM T66665 CBY5H2 10019463 IC50 = 20000 nM T66665 CTR6H1 10019555 IC50 = 38 nM T66665 CLEY67 10019929 IC50 = 1500 nM T66665 CC7M1T 10020588 IC50 = 31.6 nM T66665 CY4K1P 10021211 IC50 = 4786.3 nM T66665 C3Y6TP 10021497 IC50 = 0.09 nM T66665 C05TFO 10021647 IC50 = 9 nM T66665 CG49LP 10021928 IC50 = 45000 nM T66665 CQH70M 10022177 IC50 = 65000 nM T66665 C0UN1I 10022305 IC50 = 21000 nM T66665 CC03QH 10024599 IC50 = 20 nM T66665 CPVJ72 10024894 IC50 = 30 nM T66665 C0GC4S 10027372 IC50 = 5000 nM T66665 C7IEL6 10037656 IC50 = 300 nM T66665 CDE7V9 10038859 IC50 = 290 nM T66665 C4CD3P 10040599 IC50 = 120000 nM T66665 C1EAZ3 10041271 IC50 = 90 nM T66665 CI6F3U 10044786 IC50 = 1.68 nM T66665 CIS0T3 10046006 IC50 = 60 nM T66665 C9C4IM 10046378 IC50 = 1.995 nM T66665 C71ION 10047011 IC50 = 35500 nM T66665 CT54KN 10047220 IC50 = 11200 nM T66665 CH4F5X 10050648 IC50 = 592 nM T66665 CRK0M8 10051539 IC50 = 1000 nM T66665 C8WTM1 10064144 IC50 = 3 nM T66665 CS40HT 10064410 IC50 = 34000 nM T66665 CT1VG7 10067604 IC50 = 500 nM T66665 C58CDE 10068193 IC50 = 650 nM T66665 C7U9DB 10069246 IC50 = 120 nM T66665 CCP45I 10070193 IC50 = 960 nM T66665 CY16VM 10071460 IC50 = 20 nM T66665 C5WE9A 10071673 IC50 = 300000 nM T66665 C1AV9L 10076665 IC50 > 300000 nM T66665 CJN53X 10084869 IC50 = 196 nM T66665 CSA7R2 10088207 IC50 = 40 nM T66665 CCQ28U 10088506 IC50 = 500 nM T66665 CW05LQ 10090654 IC50 = 1.26 nM T66665 CEX30I 10091264 IC50 = 146 nM T66665 C54JLZ 10093810 IC50 = 70 nM T66665 C9HR8U 10095369 IC50 = 67 nM T66665 C7IEF9 10095474 IC50 = 3700 nM T66665 C74OAD 10097252 IC50 > 300000 nM T66665 CHV67O 10108931 IC50 = 300 nM T66665 C92OBR 10109075 IC50 = 830 nM T66665 CW3J9B 10109361 IC50 = 940 nM T66665 C90KPZ 10109982 IC50 = 39 nM T66665 CF2L8T 10110298 IC50 = 60.26 nM T66665 C67SQN 10110427 IC50 = 338.84 nM T66665 CRKC39 10110822 IC50 = 180 nM T66665 C94UAS 10112273 IC50 = 23.99 nM T66665 CO98VP 10113620 IC50 = 7 nM T66665 CIF46A 10118686 IC50 = 480 nM T66665 C0QF5M 10131479 IC50 = 5 nM T66665 CBDU01 10133653 IC50 = 75 nM T66665 CU2TS5 10133741 IC50 = 170 nM T66665 CPEL28 10133748 IC50 = 70 nM T66665 CFX3A1 10134234 IC50 = 10000 nM T66665 C64UXL 10134425 IC50 = 40 nM T66665 CO0EY4 10134426 IC50 = 30 nM T66665 CL4ZX6 10135355 IC50 = 15.85 nM T66665 CUC48F 10136509 IC50 = 150 nM T66665 C62HSP 10138952 IC50 = 150 nM T66665 C39FVT 10154719 IC50 = 120 nM T66665 C3ALT5 10155221 IC50 = 4 nM T66665 CU0QS9 10155469 IC50 = 7 nM T66665 CCFX37 10155819 IC50 = 39.81 nM T66665 CXL35F 10156006 IC50 = 800 nM T66665 C89SFQ 10156048 IC50 = 83.18 nM T66665 CGY3U6 10156369 IC50 = 20 nM T66665 C75HBA 10156402 IC50 = 6 nM T66665 CYXL62 10156660 IC50 = 69 nM T66665 CY8WB7 10156700 IC50 = 8 nM T66665 C97MLG 10156720 IC50 = 436.52 nM T66665 CT16EK 10157135 IC50 = 17 nM T66665 C0LZU6 10157427 IC50 < 10 nM T66665 C8EP6N 10157624 IC50 = 8 nM T66665 C91PJR 10157862 IC50 = 23 nM T66665 CB8PS0 10158806 IC50 = 3 nM T66665 CN62VZ 10159879 IC50 = 19.95 nM T66665 CG6FC7 10172237 IC50 = 110 nM T66665 C3EFY5 10177578 IC50 = 7 nM T66665 CE9PV5 10177830 IC50 = 16 nM T66665 CP3C8N 10177845 IC50 = 1800 nM T66665 C1O8JD 10178729 IC50 = 1 nM T66665 C4U5VF 10179720 IC50 = 13 nM T66665 CPTS56 10179876 IC50 = 7 nM T66665 C50MBD 10180742 IC50 = 0.28 nM T66665 C73DEB 10181405 IC50 = 8230 nM T66665 CK05GP 10183636 IC50 = 310 nM T66665 CG2Y1Q 10199429 IC50 = 1500 nM T66665 C9VW0L 10199643 IC50 = 90 nM T66665 C5WB6K 10199764 IC50 = 158.49 nM T66665 CN5O6D 10199832 IC50 = 109.65 nM T66665 C7V6HN 10200639 IC50 = 40 nM T66665 COEJ03 10200640 IC50 = 20 nM T66665 CT4I3O 10200696 IC50 = 25 nM T66665 CZL86N 10200745 IC50 = 20 nM T66665 C10MGH 10200861 IC50 = 109.65 nM T66665 CXA45O 10200928 IC50 = 30 nM T66665 CBD58L 10201258 IC50 = 190.11 nM T66665 C5GSU9 10201259 IC50 = 239.99 nM T66665 CLI4G2 10201726 IC50 = 2630 nM T66665 C0CDF4 10201744 IC50 = 100 nM T66665 CIG42D 10202758 IC50 = 600 nM T66665 CS4Y1F 10221647 IC50 = 200 nM T66665 C0E4ZO 10221859 IC50 = 60.01 nM T66665 C12ZGN 10222021 IC50 > 10000 nM T66665 CW17QB 10222707 IC50 = 56 nM T66665 C1OH3T 10222861 IC50 = 80 nM T66665 C74EPI 10223326 IC50 = 28 nM T66665 C6JLS5 10223461 IC50 = 33 nM T66665 CEKL34 10224978 IC50 = 15 nM T66665 CK31YH 10224979 IC50 = 56 nM T66665 CCT79E 10227082 IC50 = 440 nM T66665 C9CX4E 10236948 IC50 = 0.09 nM T66665 CRF02L 10246625 IC50 = 500 nM T66665 C50FGR 10247267 IC50 = 42000 nM T66665 C9Q3GN 10251114 IC50 = 60 nM T66665 C1YF7W 10255326 IC50 = 1060 nM T66665 C1R9VI 10265882 IC50 = 2800 nM T66665 COQ0I9 10267703 IC50 = 18 nM T66665 CRVU30 10268555 IC50 = 3 nM T66665 C5U6ZL 10269056 IC50 = 68 nM T66665 COG84H 10269175 IC50 = 15.85 nM T66665 CDJO97 10269858 IC50 = 23 nM T66665 C4D1AW 10270798 IC50 = 100 nM T66665 CRP52C 10271231 IC50 = 416.87 nM T66665 CKZ72U 10271396 IC50 = 58 nM T66665 CNJ96H 10272113 IC50 = 290 nM T66665 CU45JL 10272435 IC50 = 10 nM T66665 CQ6ZK8 10273159 IC50 = 9 nM T66665 C15AKU 10273161 IC50 > 10000 nM T66665 CVQ9R1 10273329 IC50 = 21 nM T66665 CCT59Q 10273651 IC50 = 530 nM T66665 CA5FY9 10286243 IC50 = 18520 nM T66665 CJE46B 10292387 IC50 = 52.48 nM T66665 CV2OS0 10292572 IC50 = 1349.9 nM T66665 C3GB8J 10292693 IC50 = 50 nM T66665 C19RZV 10293184 IC50 = 2884.03 nM T66665 CG1I7N 10293242 IC50 = 288.4 nM T66665 C8AFM7 10293899 IC50 = 1300 nM T66665 CX3J6F 10294269 IC50 = 5 nM T66665 CA37EH 10294458 IC50 = 6 nM T66665 CYW2V3 10294501 IC50 = 120 nM T66665 C9JN8Q 10294921 IC50 = 239.88 nM T66665 CR02XQ 10295072 IC50 = 7 nM T66665 C2QA8P 10296709 IC50 = 5.3 nM T66665 C38RAI 10313600 IC50 = 12670 nM T66665 C5AN4G 10316456 IC50 = 63000 nM T66665 C7JIZ5 10316538 IC50 = 34500 nM T66665 C3X7IN 10316629 IC50 = 3.981 nM T66665 CK1WP4 10316962 IC50 = 17500 nM T66665 CJ6RY9 10317408 IC50 = 1.459 nM T66665 C1OSM9 10318787 IC50 < 10 nM T66665 CITV57 10319221 IC50 = 900 nM T66665 C1C4NS 10330671 IC50 = 16500 nM T66665 C1LZ7Y 10335263 IC50 = 30 nM T66665 CWG32C 10336743 IC50 = 9705.1 nM T66665 CB06KL 10336873 IC50 = 250 nM T66665 C7AY2L 10337564 IC50 = 3000 nM T66665 CCV82I 10339513 IC50 = 18000 nM T66665 CA3XB0 10339727 IC50 = 51.29 nM T66665 CD39QI 10340792 IC50 = 25000 nM T66665 CY6D5M 10342564 IC50 = 88000 nM T66665 C1REP8 10355223 IC50 > 100000 nM T66665 CLID50 10359269 IC50 = 4800 nM T66665 CM01BR 10359484 IC50 = 200 nM T66665 C6P9HD 10360345 IC50 = 6 nM T66665 CJG7W4 10360688 IC50 = 758.58 nM T66665 C8IJG9 10361245 IC50 = 970 nM T66665 CVCX96 10362126 IC50 = 0.17 nM T66665 CE19XH 10362365 IC50 = 130 nM T66665 CX3C0N 10362509 IC50 = 33.5 nM T66665 CI42KJ 10363144 IC50 = 10 nM T66665 CL41EY 10363199 IC50 = 40000 nM T66665 CX8ZA1 10363491 IC50 = 20 nM T66665 CAB38Y 10365186 IC50 = 8.356 nM T66665 CR5JS6 10369485 IC50 = 7 nM T66665 CKH1A6 10381453 IC50 = 18879.91 nM T66665 C9CJY4 10381501 IC50 = 100 nM T66665 CH8WQ5 10381921 IC50 = 4.2 nM T66665 CDB2Z0 10383075 IC50 = 43 nM T66665 C7VP2Q 10385170 IC50 = 199.53 nM T66665 CI67YJ 10385715 IC50 = 12 nM T66665 C9SPO1 10385880 IC50 = 13 nM T66665 CY4W2C 10386019 IC50 = 12 nM T66665 C0XNA3 10389320 IC50 = 40 nM T66665 CSR51N 10403254 IC50 = 3 nM T66665 CA7QF5 10405126 IC50 = 6606.93 nM T66665 CFL72P 10405693 IC50 = 120 nM T66665 CW83GT 10406349 IC50 = 0.06998 nM T66665 C5JHI0 10406427 IC50 = 1800 nM T66665 CFXL12 10406946 IC50 = 3.5 nM T66665 CP40MA 10407440 IC50 = 4 nM T66665 C17TBC 10407720 IC50 = 100 nM T66665 C9SRX6 10408088 IC50 = 14 nM T66665 C39ISW 10408494 IC50 = 5 nM T66665 CFK2J0 10409583 IC50 = 66000 nM T66665 C52MXI 10413126 IC50 = 38400 nM T66665 CT16GY 10413362 IC50 = 8200 nM T66665 C2L8RQ 10424013 IC50 > 30000 nM T66665 CA3X7E 10424186 IC50 > 100000 nM T66665 CA1S7I 10425292 IC50 = 46 nM T66665 CGU4Q8 10425834 IC50 = 510 nM T66665 CW6H4S 10426661 IC50 = 3200 nM T66665 CP57LS 10426884 IC50 = 80 nM T66665 CQ7Z6C 10428486 IC50 = 5100 nM T66665 CL15GH 10429020 IC50 = 1000 nM T66665 CJIO54 10429739 IC50 = 0.005998 nM T66665 C3NK6J 10430343 IC50 = 520 nM T66665 CJNV54 10431739 IC50 = 298200 nM T66665 CA24ER 10433546 IC50 = 50 nM T66665 C1T4PM 10446327 IC50 > 30000 nM T66665 C65BPM 10447425 IC50 = 2250 nM T66665 C72ERI 10448879 IC50 = 77900 nM T66665 CIMC74 10449604 IC50 = 260 nM T66665 CA9PQ4 10449908 IC50 = 64400 nM T66665 CXB21M 10452212 IC50 = 0.02 nM T66665 CVF6I8 10452350 IC50 = 790 nM T66665 CLV8C6 10452657 IC50 = 7730 nM T66665 CQ94JT 10453591 IC50 = 22 nM T66665 CGD93Y 10457034 IC50 = 40 nM T66665 C1WM2V 10459826 IC50 = 45 nM T66665 CB50TO 10471014 IC50 = 14.13 nM T66665 C4TMQ6 10471276 IC50 = 300 nM T66665 CJ4T9S 10472587 IC50 = 3500 nM T66665 C3TK7X 10472597 IC50 = 1550 nM T66665 C9DB6Y 10474426 IC50 = 72000 nM T66665 C7DT1E 10476542 IC50 < 10 nM T66665 CX8BU5 10476854 IC50 = 50 nM T66665 COL4Z0 10476930 IC50 = 30 nM T66665 CXE0V2 10482075 IC50 = 1 nM T66665 CUP86R 10490919 IC50 > 40000 nM T66665 CLP06F 10493616 IC50 = 40 nM T66665 C3ZM1X 10494600 IC50 = 90 nM T66665 C82ILQ 10497855 IC50 = 3000 nM T66665 CMS87O 10497881 IC50 = 28 nM T66665 C4CRG9 10498736 IC50 = 21.88 nM T66665 C5CZB7 10498979 IC50 = 1129.8 nM T66665 CHQ85J 10499452 IC50 > 100000 nM T66665 CI0S4Q 10499717 IC50 > 10000 nM T66665 CZD6A8 10500038 IC50 = 5754.4 nM T66665 CW9EQ6 10500466 IC50 = 12.02 nM T66665 CC0Z4F 10500696 IC50 = 300 nM T66665 CPO37N 10500778 IC50 = 1 nM T66665 CZ7IX5 10500888 IC50 = 1470 nM T66665 C65HEP 10501037 IC50 = 109.65 nM T66665 CMJ08V 10501190 IC50 = 109.65 nM T66665 C1J3DI 10501213 IC50 > 10000 nM T66665 CU8KR5 10501652 IC50 = 707.95 nM T66665 C6O1UH 10501957 IC50 = 30 nM T66665 C2QN6Y 10501958 IC50 = 79.43 nM T66665 CE4S1Y 10502827 IC50 = 19.95 nM T66665 CGB5H6 10504452 IC50 = 1000 nM T66665 CQ6RL5 10504460 IC50 = 50 nM T66665 CR4OK6 10504537 IC50 = 30 nM T66665 CB84IP 10505250 IC50 > 66000 nM T66665 CI16BX 10506935 IC50 = 90 nM T66665 C9L8JW 10514848 IC50 > 40000 nM T66665 CMF9R3 10516041 IC50 > 50000 nM T66665 CI6F7S 10516483 IC50 = 95 nM T66665 C3ZL6Y 10517042 IC50 > 40000 nM T66665 CCO02A 10517413 IC50 = 550 nM T66665 C8JTN1 10518222 IC50 = 1870 nM T66665 CGC62Z 10519259 IC50 = 47100 nM T66665 C80QLC 10519522 IC50 = 9500 nM T66665 CF57BP 10520447 IC50 > 100000 nM T66665 CO6D8P 10520508 IC50 = 199.53 nM T66665 C9WDP7 10520866 IC50 = 640 nM T66665 CHCD84 10521129 IC50 > 10000 nM T66665 CZ4MX2 10521318 IC50 = 90 nM T66665 CL2WV6 10521660 IC50 = 14 nM T66665 CLK73W 10521710 IC50 = 4000 nM T66665 CLZ4D8 10522463 IC50 = 52300 nM T66665 CGMA31 10522592 IC50 = 3 nM T66665 CS3L6E 10522977 IC50 = 150 nM T66665 CQ3S6J 10523033 IC50 = 2 nM T66665 C35MKT 10523190 IC50 = 61.66 nM T66665 CCM67S 10523255 IC50 = 1621.81 nM T66665 CB2EZ0 10523413 IC50 = 19 nM T66665 C7C0WZ 10523638 IC50 > 10000 nM T66665 CXO9S1 10524261 IC50 > 100000 nM T66665 C52QXF 10524370 IC50 = 3.981 nM T66665 CU7Z4M 10524532 IC50 = 470 nM T66665 C17KQI 10524587 IC50 = 12.88 nM T66665 C0N4YM 10524857 IC50 = 80 nM T66665 CA4TO8 10524898 IC50 > 100000 nM T66665 CEO49Q 10524951 IC50 > 100000 nM T66665 CS14IM 10525575 IC50 = 192 nM T66665 CTKM86 10525659 IC50 = 1090 nM T66665 CRI9N3 10526696 IC50 > 100000 nM T66665 CF1PX9 10526904 IC50 > 100000 nM T66665 CH1FP4 10528852 IC50 > 8000 nM T66665 CX0WN5 10535894 IC50 > 1000000 nM T66665 CEG9B5 10536723 IC50 = 360000 nM T66665 CDBH49 10539507 IC50 > 40000 nM T66665 CL8SI7 10539571 IC50 > 40000 nM T66665 C54DWE 10541466 IC50 = 4500 nM T66665 C8YI0Q 10541610 IC50 > 100000 nM T66665 C58BNM 10543451 IC50 = 5200 nM T66665 CN6M2J 10543472 IC50 = 4500 nM T66665 CNQ03M 10544389 IC50 = 790 nM T66665 CU8TZ2 10544709 IC50 = 1000 nM T66665 CUAQ98 10545165 IC50 = 26000 nM T66665 C4AV8Q 10545354 IC50 = 6 nM T66665 C47RFN 10545379 IC50 = 1559.55 nM T66665 CIB05E 10545620 IC50 = 100 nM T66665 C4N8QO 10545724 IC50 = 20700 nM T66665 C9UB1K 10546170 IC50 > 100000 nM T66665 CQ32BJ 10546382 IC50 = 3890.45 nM T66665 C0JP5I 10546567 IC50 = 14 nM T66665 C1TPD4 10547228 IC50 = 1540 nM T66665 C2YV6X 10547351 IC50 = 5 nM T66665 C8MGI2 10548394 IC50 > 10000 nM T66665 C8U3CE 10548520 IC50 = 20.89 nM T66665 CICG32 10549411 IC50 = 19.95 nM T66665 C1H7JD 10549466 IC50 = 20.89 nM T66665 CBH0K1 10549551 IC50 = 575.44 nM T66665 C62ITD 10549657 IC50 > 100000 nM T66665 C1YLO7 10549795 IC50 = 6 nM T66665 CU4WD3 10551821 IC50 = 60 nM T66665 C1Q9ZA 10552224 IC50 = 47 nM T66665 C56IOS 10563335 IC50 = 510000 nM T66665 CIR1X4 10563380 IC50 = 3500 nM T66665 CCNY05 10564674 IC50 > 100000 nM T66665 C6M5YN 10567176 IC50 = 1530 nM T66665 C9SOC2 10568310 IC50 = 3000 nM T66665 CP6JX9 10568417 IC50 > 100000 nM T66665 CM89NX 10569712 IC50 = 750 nM T66665 CU1RH9 10569839 IC50 = 1819.7 nM T66665 CG8HY7 10569949 IC50 = 100 nM T66665 CS74PE 10570051 IC50 = 2900 nM T66665 CU5GB2 10570135 IC50 = 5 nM T66665 CN2W5O 10570444 IC50 = 170 nM T66665 CZAS51 10570709 IC50 = 100 nM T66665 CZ38CW 10570970 IC50 > 100000 nM T66665 C6FAO5 10571335 IC50 = 10 nM T66665 CN1TG0 10571627 IC50 = 1.995 nM T66665 C9PT5C 10571870 IC50 = 54000 nM T66665 CGVM06 10572070 IC50 = 100 nM T66665 CLBY56 10572128 IC50 = 10 nM T66665 CADV12 10572129 IC50 = 30 nM T66665 CQAJ45 10572620 IC50 = 6 nM T66665 C5WPQ6 10573666 IC50 = 9.333 nM T66665 CYJ9V0 10574324 IC50 = 3.981 nM T66665 CX17PF 10574332 IC50 = 12200 nM T66665 C5HXO6 10574480 IC50 = 330 nM T66665 CUY9N4 10574542 IC50 > 100000 nM T66665 C1ECI8 10574823 IC50 = 1.995 nM T66665 CE98XT 10574865 IC50 = 50 nM T66665 CB1ZN7 10575085 IC50 = 120 nM T66665 C6LSX4 10575260 IC50 = 323.59 nM T66665 CDA0F5 10575436 IC50 = 20.89 nM T66665 CHM8O7 10576610 IC50 = 140 nM T66665 CQ6N1V 10576818 IC50 = 5000 nM T66665 C2P3EL 10576988 IC50 = 50 nM T66665 CKXU49 10577339 IC50 = 45 nM T66665 C3P8XQ 10590357 IC50 > 30000 nM T66665 C2UPC7 10592313 IC50 = 440 nM T66665 C3ZQ9G 10592466 IC50 = 1.995 nM T66665 C0PNH9 10592721 IC50 = 400 nM T66665 CQ5HY9 10594681 IC50 = 3.3 nM T66665 CD53SH 10594762 IC50 = 100 nM T66665 CI6WX3 10594776 IC50 > 100000 nM T66665 CEH6S3 10594921 IC50 = 17 nM T66665 CV61CE 10594959 IC50 = 2000 nM T66665 C32XIL 10595453 IC50 = 22.91 nM T66665 CF8JP2 10596233 IC50 = 169.82 nM T66665 CH7V5Q 10596355 IC50 > 10000 nM T66665 C48WTA 10596725 IC50 = 3.02 nM T66665 C9S6WU 10596883 IC50 = 100000 nM T66665 CTO61I 10597216 IC50 = 338.84 nM T66665 CR9D4F 10597571 IC50 = 134.9 nM T66665 C23IOF 10598294 IC50 = 7.943 nM T66665 CY29BU 10598409 IC50 = 724.44 nM T66665 CN03KT 10598578 IC50 = 3.7 nM T66665 C8DT5Q 10598702 IC50 = 660 nM T66665 CE6TN2 10599548 IC50 > 66000 nM T66665 CCY5L1 10600544 IC50 = 30 nM T66665 CSH85U 10600655 IC50 = 140 nM T66665 CW8G7F 10600662 IC50 = 30.2 nM T66665 CG3YV0 10600758 IC50 = 300 nM T66665 CUZ7B1 10615540 IC50 = 400 nM T66665 CT5S2N 10616370 IC50 = 2500 nM T66665 CG2A5Z 10616776 IC50 = 18 nM T66665 C37IWY 10617890 IC50 = 1499.68 nM T66665 C8YQ6N 10618038 IC50 = 3290 nM T66665 CWN28D 10618802 IC50 = 9 nM T66665 C8KLQ0 10619035 IC50 = 2.512 nM T66665 C5GWB7 10619274 IC50 = 51000 nM T66665 CV5WA8 10619336 IC50 = 70 nM T66665 C49FXO 10619703 IC50 = 79.43 nM T66665 CH4M5Z 10619979 IC50 > 10000 nM T66665 CQY85C 10620079 IC50 = 18000 nM T66665 C3U7ME 10620295 IC50 = 426.58 nM T66665 CJ8X1M 10620528 IC50 = 2 nM T66665 CEF30U 10620563 IC50 = 320 nM T66665 C8T6QN 10620570 IC50 = 33.11 nM T66665 CGN4X1 10620694 IC50 = 912.01 nM T66665 C27RKQ 10621114 IC50 > 100000 nM T66665 CX34BP 10621294 IC50 = 64.57 nM T66665 CSMA50 10621472 IC50 = 3200 nM T66665 CP63ZJ 10621562 IC50 = 140 nM T66665 CGV75S 10621593 IC50 = 19800 nM T66665 CRXA24 10621689 IC50 = 26.92 nM T66665 C0I4UK 10622186 IC50 = 346.74 nM T66665 C7Z3AE 10623138 IC50 = 1040 nM T66665 C6Z3DW 10623232 IC50 = 66 nM T66665 C8C2XD 10623316 IC50 = 10 nM T66665 CD51RW 10623882 IC50 = 60 nM T66665 C9NQP1 10624176 IC50 = 80 nM T66665 CZMB47 10624367 IC50 > 17000 nM T66665 CS37XW 10624880 IC50 = 80 nM T66665 CS5L3I 10636972 IC50 > 1000000 nM T66665 C5N1ZT 10637982 IC50 > 100000 nM T66665 CXJN98 10638180 IC50 = 220 nM T66665 C5OIE6 10639657 IC50 = 50 nM T66665 C5QJT8 10641092 IC50 = 140 nM T66665 C2H9QZ 10641380 IC50 = 251.19 nM T66665 C08ESX 10641720 IC50 > 100000 nM T66665 CJIL86 10642557 IC50 = 15 nM T66665 CB63LQ 10642954 IC50 = 4150 nM T66665 CYWU12 10643086 IC50 = 1.995 nM T66665 CV01MH 10643308 IC50 > 100000 nM T66665 CZTA61 10643309 IC50 = 14000 nM T66665 CS9X7O 10643550 IC50 = 267 nM T66665 CLZ52N 10643725 IC50 = 1999.86 nM T66665 COV2G1 10643865 IC50 = 3600 nM T66665 C6X3QR 10644259 IC50 = 10 nM T66665 CMA47V 10644309 IC50 = 3 nM T66665 C4KF7S 10644380 IC50 = 240 nM T66665 C5E1UO 10644539 IC50 = 340 nM T66665 CP9O6S 10644759 IC50 = 10 nM T66665 C0Z2LW 10645180 IC50 = 128.82 nM T66665 C3DJ8A 10645484 IC50 > 100000 nM T66665 C4I8CE 10646043 IC50 = 52.48 nM T66665 C7PXD1 10646457 IC50 = 400 nM T66665 C0EAM8 10646465 IC50 = 208.93 nM T66665 CE98OM 10646723 IC50 = 229.09 nM T66665 CV4BQ3 10647263 IC50 = 120 nM T66665 C09QKH 10648828 IC50 > 66000 nM T66665 CGO89K 10660176 IC50 > 100000 nM T66665 C97EIF 10660419 IC50 > 40000 nM T66665 C9N8EC 10662676 IC50 > 1000 nM T66665 C2UCE6 10663006 IC50 = 79000 nM T66665 C2X9JN 10663080 IC50 = 29700 nM T66665 CG9VC6 10663833 IC50 = 40 nM T66665 C6Z5MJ 10664116 IC50 > 100000 nM T66665 C4JQH6 10664141 IC50 = 4000 nM T66665 C7UP6J 10664368 IC50 > 10000 nM T66665 C65CUY 10664448 IC50 = 51.29 nM T66665 CF7I3B 10664738 IC50 = 75.86 nM T66665 CRD7N4 10665073 IC50 = 1.995 nM T66665 CMZW27 10665242 IC50 = 209.89 nM T66665 CN1I8K 10665362 IC50 = 87 nM T66665 C08GOU 10665504 IC50 > 100000 nM T66665 CCB67N 10666170 IC50 = 3.981 nM T66665 C94OSF 10666215 IC50 > 100000 nM T66665 CYU03I 10666285 IC50 > 100000 nM T66665 CN58GZ 10666572 IC50 = 4698.94 nM T66665 CX92LU 10666704 IC50 = 64700 nM T66665 CP1H7C 10667040 IC50 = 11400 nM T66665 CQUE64 10667216 IC50 = 5 nM T66665 CTY5Z0 10667341 IC50 = 1.514 nM T66665 C2B4UE 10667766 IC50 = 399.94 nM T66665 CBU0Z6 10667777 IC50 = 1.7 nM T66665 C63ZDJ 10668272 IC50 = 46800 nM T66665 CF39UA 10668540 IC50 = 169.82 nM T66665 C5BL8W 10668860 IC50 = 30 nM T66665 CQ8G9S 10668927 IC50 = 338.84 nM T66665 C72XSN 10669268 IC50 = 68100 nM T66665 C8R1WI 10669397 IC50 = 30.9 nM T66665 C3AIJ5 10669481 IC50 = 42500 nM T66665 C0L1YR 10669511 IC50 = 89.13 nM T66665 CO7MC2 10670044 IC50 > 100000 nM T66665 CC9KU0 10670425 IC50 = 1023.29 nM T66665 CF4ZD1 10670953 IC50 = 5700 nM T66665 C6CS5M 10671076 IC50 = 338.84 nM T66665 CR2WL6 10675017 IC50 = 600 nM T66665 CV0NQ2 10685244 IC50 > 40000 nM T66665 CW0M4E 10685712 IC50 = 200 nM T66665 CKZ6D7 10686987 IC50 = 520 nM T66665 C5OA4S 10688075 IC50 = 660 nM T66665 C5NZ4I 10688742 IC50 > 100000 nM T66665 CF5XO3 10688810 IC50 > 100000 nM T66665 CRWF25 10689255 IC50 = 1348.96 nM T66665 C7IMK5 10689263 IC50 > 200 nM T66665 CIMT60 10689279 IC50 = 1000 nM T66665 CIL0X1 10690090 IC50 > 10000 nM T66665 C2R0UI 10690316 IC50 = 4201 nM T66665 CA9B7R 10690364 IC50 = 45600 nM T66665 CS4QA8 10690636 IC50 = 407.38 nM T66665 C9DUH1 10691290 IC50 = 724.44 nM T66665 C58BDY 10691358 IC50 = 1999.86 nM T66665 CHO5U6 10692230 IC50 = 8.913 nM T66665 C6LDV7 10692403 IC50 = 891.25 nM T66665 C02IYT 10692761 IC50 = 30.9 nM T66665 CX93TR 10693268 IC50 = 1698.24 nM T66665 C6YVW5 10693269 IC50 = 630 nM T66665 CI9CB2 10693380 IC50 = 1096.48 nM T66665 CPZB30 10693561 IC50 = 40 nM T66665 C8W4VO 10693792 IC50 = 50 nM T66665 CPU6N3 10694708 IC50 = 40 nM T66665 CX65EM 10695000 IC50 = 29 nM T66665 CF4G6H 10708915 IC50 = 2360 nM T66665 CDPT71 10709447 IC50 = 1000 nM T66665 C1WR8U 10710181 IC50 = 45 nM T66665 CLK87B 10710312 IC50 = 62800 nM T66665 C7HT2G 10710438 IC50 > 100000 nM T66665 CQOD76 10710474 IC50 = 300 nM T66665 CE6L3I 10711484 IC50 = 510 nM T66665 CT78PA 10711485 IC50 = 1798.87 nM T66665 CFAO45 10712340 IC50 = 20.89 nM T66665 CX5I9C 10712958 IC50 = 2300 nM T66665 CCL9Z5 10712963 IC50 = 1000 nM T66665 CJR8V5 10713528 IC50 = 51 nM T66665 CBM05Q 10714139 IC50 = 100 nM T66665 C56ECJ 10714428 IC50 = 29700 nM T66665 CU20OI 10714590 IC50 = 1.995 nM T66665 CWK7C1 10714907 IC50 = 51000 nM T66665 C7IVL5 10715163 IC50 = 2600 nM T66665 C54WCH 10715239 IC50 = 933.25 nM T66665 C03QYS 10715523 IC50 > 100000 nM T66665 CEZK47 10715707 IC50 = 2133 nM T66665 CE7M6G 10716372 IC50 = 26 nM T66665 CSHM17 10716420 IC50 = 19 nM T66665 CAZ14N 10716484 IC50 = 467.74 nM T66665 C89XSQ 10717305 IC50 = 158.49 nM T66665 C2ICZ5 10717364 IC50 > 100000 nM T66665 CUL45S 10718261 IC50 > 66000 nM T66665 CO89KL 10729633 IC50 > 50000 nM T66665 CB0A2M 10729933 IC50 = 8000 nM T66665 CE4GJ6 10734248 IC50 = 4660 nM T66665 CZD32K 10735037 IC50 > 100000 nM T66665 CLQ29C 10737761 IC50 = 80 nM T66665 CPQ73G 10738225 IC50 = 100000 nM T66665 C8WKH3 10738721 IC50 = 3580 nM T66665 CB4Y8S 10738786 IC50 = 758.58 nM T66665 CM8DE5 10738921 IC50 = 100000 nM T66665 C2O5VB 10739009 IC50 = 12.88 nM T66665 C8Q9WG 10739510 IC50 = 570 nM T66665 CG6TM0 10739730 IC50 = 250 nM T66665 C8TQ2M 10740301 IC50 = 14300 nM T66665 C2L9KP 10740567 IC50 = 457.09 nM T66665 CFAL86 10740669 IC50 = 1200 nM T66665 CF6QR7 10741315 IC50 = 128.82 nM T66665 C4UQ2F 10741367 IC50 = 170 nM T66665 CNSW35 10741533 IC50 = 169.82 nM T66665 CCDT10 10742004 IC50 = 950 nM T66665 C14GVA 10742263 IC50 = 12 nM T66665 C79QXL 10742264 IC50 > 100000 nM T66665 CZ1R8L 10742692 IC50 = 2500 nM T66665 CORK85 10743328 IC50 = 60 nM T66665 C4JNI5 10746383 IC50 = 7500 nM T66665 CJR19I 10757665 IC50 = 38 nM T66665 C31ZYT 10758665 IC50 = 980 nM T66665 CKJB53 10758721 IC50 = 479.73 nM T66665 C41VSC 10759467 IC50 = 1.5 nM T66665 CI9LE3 10759852 IC50 = 288.4 nM T66665 CEX12Q 10759876 IC50 = 1700 nM T66665 C60QMK 10760082 IC50 > 10000 nM T66665 CE8TP5 10760536 IC50 = 2870 nM T66665 C34ECZ 10760894 IC50 = 1 nM T66665 CT9U8B 10760960 IC50 = 1 nM T66665 CW85FZ 10761459 IC50 = 10 nM T66665 CUB65A 10761664 IC50 = 83 nM T66665 CYH42G 10762072 IC50 > 100000 nM T66665 CA9Y7S 10762141 IC50 > 100000 nM T66665 CZ12TA 10762494 IC50 = 616.6 nM T66665 CBP31E 10763244 IC50 > 10000 nM T66665 C3VNE9 10763435 IC50 = 230 nM T66665 CL91JT 10764155 IC50 = 346.74 nM T66665 C43ANY 10764356 IC50 = 21.88 nM T66665 CWD6R8 10765040 IC50 = 28.18 nM T66665 CY62TN 10765111 IC50 = 26.92 nM T66665 CQ1YE3 10765731 IC50 = 80 nM T66665 C2O5CV 10765773 IC50 = 7 nM T66665 CAV79K 10766450 IC50 > 8000 nM T66665 C5TRJ4 10766544 IC50 = 40 nM T66665 CHK8S2 10766586 IC50 = 140 nM T66665 CWD23P 10776967 IC50 > 40000 nM T66665 CBX0D1 10778330 IC50 > 50000 nM T66665 C08QRP 10780700 IC50 > 1000000 nM T66665 CN0CO3 10781432 IC50 = 250 nM T66665 CWM20X 10782440 IC50 = 61 nM T66665 C6OSX7 10783363 IC50 > 10000 nM T66665 CG5EO7 10783872 IC50 = 50 nM T66665 C1SAW6 10783884 IC50 = 190 nM T66665 CT81VO 10784091 IC50 = 30.2 nM T66665 CIFQ86 10784411 IC50 = 1 nM T66665 CNB21H 10784589 IC50 = 229.09 nM T66665 CXE17N 10784741 IC50 = 330 nM T66665 CJ8BO1 10784838 IC50 = 16.98 nM T66665 CAE0J1 10786069 IC50 = 9549.93 nM T66665 C54TIZ 10786081 IC50 = 12 nM T66665 C4K0GX 10786241 IC50 > 100000 nM T66665 CE5Z1V 10786868 IC50 = 154 nM T66665 C1IZB3 10786954 IC50 = 2 nM T66665 CA9U0M 10786970 IC50 = 37600 nM T66665 C37NKS 10786971 IC50 = 6.761 nM T66665 CLD35X 10787338 IC50 = 32 nM T66665 CYRC45 10787698 IC50 = 169.82 nM T66665 C0X7ME 10787761 IC50 = 645.65 nM T66665 CL6I5P 10787918 IC50 = 954.99 nM T66665 C1LRD4 10789363 IC50 > 100000 nM T66665 C0EOC9 10791740 IC50 = 60 nM T66665 CA17RT 10799759 IC50 > 100000 nM T66665 CU80LF 10802365 IC50 = 6000 nM T66665 CM13QH 10804032 IC50 > 100000 nM T66665 CO8XJ4 10805003 IC50 = 60 nM T66665 CSYE98 10807025 IC50 = 50 nM T66665 CPYI68 10807315 IC50 > 100000 nM T66665 C32KJP 10807549 IC50 = 1800 nM T66665 C8JM6A 10808251 IC50 = 33.11 nM T66665 CPA3M7 10808453 IC50 = 59000 nM T66665 CYN31S 10808713 IC50 = 100 nM T66665 CS3L2R 10809519 IC50 = 5.012 nM T66665 C1DYX5 10809854 IC50 = 1288.25 nM T66665 C4CBE7 10809855 IC50 = 1819.7 nM T66665 C4IZ1J 10809969 IC50 > 100000 nM T66665 C1VG3L 10810038 IC50 = 398.11 nM T66665 CXEV84 10810080 IC50 > 100000 nM T66665 C2DP6S 10810285 IC50 = 2500 nM T66665 C69ZEY 10810604 IC50 = 3 nM T66665 CY65XB 10810622 IC50 = 330 nM T66665 C68IWJ 10810738 IC50 = 346.74 nM T66665 CLIV93 10810863 IC50 > 100000 nM T66665 CY4AX3 10811597 IC50 = 10 nM T66665 C41MJH 10812437 IC50 = 5.7 nM T66665 CQEP24 10812568 IC50 = 250 nM T66665 COQ40E 10812673 IC50 = 1.288 nM T66665 CF5JL0 10813070 IC50 = 60 nM T66665 CT9ND3 10813498 IC50 = 75 nM T66665 C0J9RB 10813571 IC50 = 50 nM T66665 C9X2TQ 10814249 IC50 = 680 nM T66665 CPR41W 10816219 IC50 > 100000 nM T66665 C59HAF 10829130 IC50 = 1599.56 nM T66665 CZ0C4S 10829132 IC50 = 10200 nM T66665 CE92RY 10829314 IC50 = 250 nM T66665 C50RZL 10830016 IC50 = 20000 nM T66665 CU6T5D 10830211 IC50 = 934000 nM T66665 CG9A0R 10830212 IC50 > 100000 nM T66665 C3WOM2 10830272 IC50 = 340 nM T66665 C2F1RB 10830394 IC50 = 600 nM T66665 CKY2T4 10830950 IC50 = 4000 nM T66665 C7D4TN 10831290 IC50 = 928.97 nM T66665 C56CIL 10831559 IC50 = 510 nM T66665 CCLK02 10831725 IC50 = 340 nM T66665 C2UV9K 10831758 IC50 > 10000 nM T66665 CX97QO 10832104 IC50 = 175 nM T66665 CMDL97 10832170 IC50 = 3230 nM T66665 CFXZ69 10832238 IC50 = 7 nM T66665 CSCA58 10832407 IC50 = 363.08 nM T66665 CJA96D 10832510 IC50 = 8350 nM T66665 C4JO1V 10832560 IC50 = 50 nM T66665 CS2L9C 10833127 IC50 = 120.23 nM T66665 CO8R6S 10833677 IC50 = 779.83 nM T66665 CNE4F5 10834020 IC50 = 1096.48 nM T66665 C54SBR 10834201 IC50 = 5 nM T66665 C73TZG 10834744 IC50 > 100000 nM T66665 CV9Z3G 10834794 IC50 = 100 nM T66665 CE2HY4 10835226 IC50 = 890 nM T66665 CUXE91 10835645 IC50 = 346.74 nM T66665 CTU46J 10836128 IC50 = 426.58 nM T66665 C6B8WX 10836221 IC50 = 1445.44 nM T66665 C12PJQ 10836527 IC50 = 30 nM T66665 CDJ8Y3 10847385 IC50 = 260000 nM T66665 CK2VU6 10848242 IC50 > 50000 nM T66665 CA06GJ 10850087 IC50 > 40000 nM T66665 CHZW73 10850787 IC50 = 15000 nM T66665 CF98BX 10850793 IC50 = 70 nM T66665 C3PCB0 10851091 IC50 = 150 nM T66665 CA8JU0 10851763 IC50 = 30000 nM T66665 C46JCP 10852345 IC50 = 7 nM T66665 CZI74A 10852952 IC50 > 100000 nM T66665 CIW26O 10853420 IC50 = 24400 nM T66665 CBVH56 10853804 IC50 > 100000 nM T66665 C9RQ7H 10854191 IC50 = 100 nM T66665 C92EYG 10860016 IC50 = 5380 nM T66665 C86IWR 10862599 IC50 = 13500 nM T66665 CLU6A5 10872407 IC50 > 1000 nM T66665 CWX81R 10872725 IC50 > 10000 nM T66665 C35PLX 10872752 IC50 > 10000 nM T66665 CQLZ76 10873532 IC50 = 3720 nM T66665 CB7IT1 10882387 IC50 = 51 nM T66665 C1N4JQ 10882657 IC50 = 14 nM T66665 C2JF4U 10882658 IC50 = 28 nM T66665 C3DCA9 10893410 IC50 = 3 nM T66665 C2S7FM 10893857 IC50 > 10000 nM T66665 CDHF71 10894407 IC50 = 74 nM T66665 C76DQF 10894687 IC50 > 20000 nM T66665 C5DNU3 10895294 IC50 = 34 nM T66665 C1DQ9B 10901219 IC50 = 4960 nM T66665 CF0CX3 10904046 IC50 > 1000 nM T66665 C7DR3V 10908643 IC50 > 100 ug.mL-1 T66665 CJV6C1 10914501 IC50 = 144 nM T66665 C5Y2AC 10914865 IC50 = 2630 nM T66665 COS6R7 10926603 IC50 = 6 nM T66665 CAEI48 10936484 IC50 = 20 nM T66665 CPNK84 10936619 IC50 = 19700 nM T66665 CP5W3G 10937079 IC50 = 120 nM T66665 CYSJ65 10937794 IC50 = 11 nM T66665 CD1N3J 10938268 IC50 > 1000 nM T66665 CTC5M0 10947004 IC50 > 100000 nM T66665 CSO6I1 10947517 IC50 > 100000 nM T66665 CTK81L 10948456 IC50 = 11 nM T66665 CEA2N7 10960870 IC50 > 10000 nM T66665 C1K0DF 10980892 IC50 > 10000 nM T66665 C5VRD8 10981473 IC50 = 42 nM T66665 C1RHL4 10990488 IC50 = 827 nM T66665 CT3PX2 10991144 IC50 = 13900 nM T66665 C93BPL 10991235 IC50 = 9 nM T66665 C9KIM8 10991648 IC50 = 187 nM T66665 C74RTU 10991908 IC50 > 10000 nM T66665 C5FAQ4 10992868 IC50 = 53 nM T66665 CY2J9R 11002614 IC50 > 100000 nM T66665 CS21NJ 11003065 IC50 = 600 nM T66665 CQ3M8H 11012540 IC50 > 10000 nM T66665 C24SDE 11024492 IC50 > 10000 nM T66665 CK25QF 11025137 IC50 = 51300 nM T66665 C0O4NS 11025223 IC50 = 13 nM T66665 CQK2S8 11025447 IC50 > 10000 nM T66665 CGSD64 11034312 IC50 = 36700 nM T66665 CT2CH1 11035516 IC50 = 14 nM T66665 CG4QE8 11036302 IC50 = 15 nM T66665 C5XQ9U 11036926 IC50 > 10000 nM T66665 C81NLC 11046361 IC50 > 10000 nM T66665 CMW94C 11046805 IC50 = 18 nM T66665 C1O6JT 11046829 IC50 = 43 nM T66665 C15YND 11056746 IC50 = 2000 nM T66665 C1POL2 11057066 IC50 = 700 nM T66665 C42IZS 11058188 IC50 > 20000 nM T66665 CX60IR 11058879 IC50 = 30 nM T66665 CY9UA1 11067599 IC50 > 10000 nM T66665 CE1V0L 11067992 IC50 = 16 nM T66665 CW5F0A 11068088 IC50 = 40 nM T66665 CQ8G6P 11068955 IC50 > 10000 nM T66665 C6DWG3 11069216 IC50 = 730 nM T66665 CJ3C0Q 11070151 IC50 > 20000 nM T66665 CCM59W 11078663 IC50 = 18 nM T66665 CP38KM 11079294 IC50 = 9 nM T66665 CTB97E 11079400 IC50 = 11 nM T66665 C37LKH 11089551 IC50 > 10000 nM T66665 CW13NO 11090142 IC50 = 15 nM T66665 CHK0J7 11097158 IC50 = 5380 nM T66665 C5AD1I 11099739 IC50 = 930 nM T66665 CW47TJ 11100014 IC50 > 10000 nM T66665 C75GDS 11110406 IC50 = 10000 nM T66665 CXP08O 11110905 IC50 > 10000 nM T66665 C31WGY 11112513 IC50 = 10000 nM T66665 CK57PL 11121068 IC50 = 51 nM T66665 CC35GO 11122307 IC50 > 10000 nM T66665 CFSO12 11142523 IC50 > 10000 nM T66665 C3BJP2 11146784 IC50 > 100 ug.mL-1 T66665 C4P3WN 11150512 IC50 = 120 nM T66665 CX0Q9R 11152069 IC50 = 7600 nM T66665 CXEA13 11154503 IC50 = 3380 nM T66665 C2AI8T 11155025 IC50 = 370 nM T66665 CBRW71 11156027 IC50 = 300 nM T66665 CW1M8Q 11160272 IC50 = 9400 nM T66665 C4F6YP 11163455 IC50 = 20 nM T66665 C6WLA8 11175990 IC50 > 50000 nM T66665 C3I1XG 11178642 IC50 = 1200 nM T66665 C9KX7V 11180042 IC50 = 700 nM T66665 CZQU30 11184397 IC50 > 100000 nM T66665 C7MY6G 11187835 IC50 = 209.99 nM T66665 C9J2CU 11196915 IC50 = 270 nM T66665 CZC5U3 11198846 IC50 = 1100 nM T66665 CU82SZ 11202736 IC50 = 220 nM T66665 C8H4TN 11209828 IC50 = 530 nM T66665 C9A7JE 11211517 IC50 = 4429.96 nM T66665 C9JQK4 11211879 IC50 = 250 nM T66665 CFP64S 11212674 IC50 = 30 nM T66665 CU01PR 11213050 IC50 = 900 nM T66665 CM5Z6L 11213438 IC50 = 870 nM T66665 CYX84A 11213988 IC50 = 920 nM T66665 CDH1L4 11222461 IC50 > 10000 nM T66665 C5X0IY 11222615 IC50 = 1119.95 nM T66665 C5TBH9 11231244 IC50 > 100000 nM T66665 CC8Y0G 11234177 IC50 = 979.94 nM T66665 CGF74Z 11243701 IC50 = 6550 nM T66665 CEX39T 11244379 IC50 = 270 nM T66665 CX8TA6 11255478 IC50 = 4000 nM T66665 CP6N5B 11256540 IC50 = 440 nM T66665 C7EU3W 11256603 IC50 > 100000 nM T66665 CAT7H5 11257238 IC50 = 3480 nM T66665 CD0T4Y 11259519 IC50 = 310 nM T66665 CJ2C7K 11261258 IC50 = 820 nM T66665 C6TQW2 11278070 IC50 = 26 nM T66665 C1HQ0V 11278404 IC50 = 3280 nM T66665 CTSE12 11279052 IC50 = 260 nM T66665 C4SKT7 11279733 IC50 = 1000 nM T66665 C4TM3I 11280986 IC50 = 355 nM T66665 C9EAJ5 11281693 IC50 = 2449.06 nM T66665 CY8K9F 11282341 IC50 = 740 nM T66665 C90MDA 11282890 IC50 > 10000 nM T66665 CAXV25 11291135 IC50 > 100000 nM T66665 CXH21C 11291861 IC50 = 1800 nM T66665 CYR5J9 11292742 IC50 = 199.99 nM T66665 CFN1T0 11292891 IC50 > 10000 nM T66665 C5LG8B 11293070 IC50 = 30 nM T66665 C5M6EP 11301001 IC50 = 130 nM T66665 CU3M8C 11301795 IC50 > 100000 nM T66665 C6NI5K 11301895 IC50 = 10000 nM T66665 C8ZGQ9 11302033 IC50 > 100000 nM T66665 C6L0BA 11302745 IC50 > 100000 nM T66665 CI6LW1 11313752 IC50 = 670 nM T66665 CBDY04 11313846 IC50 = 6889.7 nM T66665 C0SA8N 11314326 IC50 = 42600 nM T66665 CZF4I8 11314954 IC50 = 9000 nM T66665 C5BSC7 11316581 IC50 > 100000 nM T66665 C0NC7H 11317417 IC50 = 930 nM T66665 CF6TZ4 11329239 IC50 = 410 nM T66665 CGL2N3 11336129 IC50 = 1780 nM T66665 CLR35D 11337592 IC50 = 50 nM T66665 C8RH4F 11338802 IC50 = 680 nM T66665 CTA54I 11340629 IC50 = 410 nM T66665 C09HXJ 11340857 IC50 = 930 nM T66665 CWMK06 11350105 IC50 = 10000 nM T66665 COY06A 11359466 IC50 = 47620 nM T66665 CB8NC3 11361946 IC50 = 1200 nM T66665 C2UG5L 11372471 IC50 = 2240 nM T66665 CL7X1Z 11373641 IC50 < 34 nM T66665 C2EJ0X 11374699 IC50 = 700 nM T66665 CF4JK1 11382191 IC50 > 100000 nM T66665 CDU98V 11382825 IC50 > 100000 nM T66665 C3F9SU 11382984 IC50 > 100000 nM T66665 CA85FN 11383735 IC50 = 320 nM T66665 CR8T2S 11384636 IC50 = 180 nM T66665 CP2ID5 11386458 IC50 > 40000 nM T66665 CXJ05V 11394262 IC50 > 10000 nM T66665 C3GOD4 11395292 IC50 = 0.44 nM T66665 CHW1N4 11395839 IC50 = 1995262.31 nM T66665 C1EL8Z 11396529 IC50 = 1440 nM T66665 CGQK95 11398561 IC50 = 100 nM T66665 C1VYZ9 11404334 IC50 = 80 nM T66665 C02PEI 11415723 IC50 > 100000 nM T66665 C8LG9O 11416157 IC50 = 9690 nM T66665 CG9BL5 11417961 IC50 = 2050 nM T66665 CLC2X3 11418074 IC50 = 380 nM T66665 C6JL8U 11419147 IC50 = 359.75 nM T66665 CC8A4V 11429689 IC50 = 71 nM T66665 C1ICK8 11430770 IC50 = 570 nM T66665 C07IKF 11439406 IC50 = 1470 nM T66665 C4F5TP 11439632 IC50 = 6400 nM T66665 CDHJ18 11440364 IC50 < 10 nM T66665 C4F9NZ 11440998 IC50 = 3990.25 nM T66665 CI6AL4 11442938 IC50 = 960 nM T66665 C2P4CT 11450459 IC50 > 100000 nM T66665 C71AVE 11459907 IC50 = 5100 nM T66665 CR2WK3 11462316 IC50 = 150 nM T66665 CTAE25 11463338 IC50 > 100000 nM T66665 CSV5L3 11463339 IC50 = 2550 nM T66665 CQ7G3L 11464135 IC50 = 242 nM T66665 C8P1SR 11472579 IC50 = 90 nM T66665 C28EVY 11473814 IC50 = 9770 nM T66665 CMO65J 11474526 IC50 > 50000 nM T66665 CB17JQ 11474778 IC50 = 2590 nM T66665 CLW8V6 11474895 IC50 > 10000 nM T66665 CFKU15 11483401 IC50 = 1990 nM T66665 CTFW72 11485547 IC50 = 1480 nM T66665 C0KFS2 11485761 IC50 = 1900 nM T66665 C6H1KP 11487377 IC50 > 100000 nM T66665 CD43NT 11487702 IC50 = 450 nM T66665 CXU3T1 11487950 IC50 = 610 nM T66665 CH0X2T 11500030 IC50 < 240 nM T66665 C23SUC 11507797 IC50 = 1280 nM T66665 COQG90 11513260 IC50 = 370 nM T66665 C71QRS 11519421 IC50 = 2200 nM T66665 CZ1LE5 11526431 IC50 > 100000 nM T66665 CDA8N6 11530051 IC50 = 73 nM T66665 C68AWO 11544686 IC50 = 494300 nM T66665 CKGE25 11544925 IC50 = 74 nM T66665 CY29OV 11546127 IC50 = 1800 nM T66665 C54ZXY 11552163 IC50 = 860 nM T66665 C5YGU8 11562265 IC50 = 5200 nM T66665 CM7S6Q 11588648 IC50 > 10000 nM T66665 C7N3CF 11608668 IC50 > 100000 nM T66665 C8DB6N 11609224 IC50 = 69 nM T66665 CZ04NY 11618742 IC50 = 3200 nM T66665 CT0MJ1 11625155 IC50 = 200 nM T66665 CL34EN 11637444 IC50 > 500000 nM T66665 CIL95X 11649268 IC50 = 2200 nM T66665 C6FXD8 11649854 IC50 = 60 nM T66665 CX0TY6 11688434 IC50 > 4000 nM T66665 CIQ9A0 11693043 IC50 = 5150 nM T66665 C03NOZ 11717695 IC50 = 1258925.41 nM T66665 CZ7CS1 11725257 IC50 = 0.5998 nM T66665 CQ8XW0 11725371 IC50 = 2 nM T66665 CH2ZL7 11725645 IC50 = 30 nM T66665 C2ONQ8 11726707 IC50 = 81000 nM T66665 C6BAV8 11728199 IC50 > 20000 nM T66665 C9BL0Q 11729490 IC50 > 10000 nM T66665 CP9N3Z 11731899 IC50 = 10000 nM T66665 CU8A0P 11731997 IC50 = 36 nM T66665 CV7WN8 11731998 IC50 = 48 nM T66665 CM4K3F 11732339 IC50 = 27 nM T66665 CH8F0P 11737673 IC50 = 300 nM T66665 C8CDF0 11739083 IC50 = 120 nM T66665 CK9H3A 11740421 IC50 = 110 nM T66665 CTX0K8 11740714 IC50 = 69000 nM T66665 C31LPN 11743998 IC50 = 92300 nM T66665 CP1MG8 11744262 IC50 = 66000 nM T66665 CU28LA 11749849 IC50 = 13840 nM T66665 CCF43X 11750118 IC50 = 60 nM T66665 CLRF90 11755350 IC50 = 12 nM T66665 C0DGK3 11757822 IC50 = 190 nM T66665 C18WRI 11759902 IC50 = 65 nM T66665 C69TMU 11759943 IC50 = 26 nM T66665 C5XM3U 11760393 IC50 = 7 nM T66665 C7CU9F 11761076 IC50 > 10000 nM T66665 C43QRI 11772569 IC50 = 1530 nM T66665 C5YRB8 11774557 IC50 = 16 nM T66665 C8RG2P 11779569 IC50 = 3.5 nM T66665 C70YSD 11783741 IC50 = 4 nM T66665 CDPH16 11791745 IC50 = 9000 nM T66665 CJRD74 11792200 IC50 = 6500 nM T66665 CPJA32 11792223 IC50 > 100000 nM T66665 C12XFM 11792433 IC50 = 758.58 nM T66665 C3QOZ8 11792902 IC50 = 1584.89 nM T66665 C5MUO6 11793188 IC50 = 407.38 nM T66665 C5HN3X 11793632 IC50 = 467.74 nM T66665 C8UZS4 11793960 IC50 > 100000 nM T66665 C82BSG 11793963 IC50 = 3715.35 nM T66665 CPMF06 11794210 IC50 = 524.81 nM T66665 CW73EF 11794212 IC50 = 5888.44 nM T66665 CT29JD 11794221 IC50 = 504 nM T66665 CUB83Z 11794411 IC50 = 5850 nM T66665 CKS37H 11794412 IC50 = 120 nM T66665 CZQU12 11795080 IC50 = 16.98 nM T66665 CW96FD 11795129 IC50 > 100000 nM T66665 C8TI9K 11795549 IC50 = 5700 nM T66665 C3G8OL 11795928 IC50 = 70000 nM T66665 CO5Y9J 11795942 IC50 = 158.49 nM T66665 C1YXB9 11796738 IC50 > 100000 nM T66665 C9O6SQ 11797537 IC50 = 20.89 nM T66665 C8R7HN 11797837 IC50 = 25.7 nM T66665 C75MBI 11797883 IC50 = 250 nM T66665 CVT0F8 11808877 IC50 = 400 nM T66665 CL28AI 11809792 IC50 = 12 nM T66665 CQU0Z5 11810629 IC50 > 10000 nM T66665 CLW72J 11823443 IC50 = 971 nM T66665 CG9NH0 11823791 IC50 = 123 nM T66665 C48YQU 11825301 IC50 > 10000 nM T66665 CK1F5U 11825947 IC50 > 10000 nM T66665 C0Y1KG 11853319 IC50 = 280 nM T66665 CO2TH7 11853321 IC50 = 700 nM T66665 C6P4KS 11853563 IC50 = 1100 nM T66665 C1ZAM7 11853569 IC50 = 3500 nM T66665 CVO72K 11853818 IC50 = 26300 nM T66665 C8K3DI 11853821 IC50 = 5800 nM T66665 CT7A0W 11853822 IC50 = 1200 nM T66665 CWCQ07 11854077 IC50 > 10000 nM T66665 C2KO9U 11854078 IC50 > 100000 nM T66665 CY78NP 11854079 IC50 > 100000 nM T66665 CO86TN 11854082 IC50 = 10000 nM T66665 CG3WU6 11854340 IC50 = 1200 nM T66665 C2YRM5 11856982 IC50 = 3000 nM T66665 CD68SB 11856984 IC50 = 4100 nM T66665 C38KZG 11978565 IC50 > 10 nM T66665 C1AOP8 11978570 IC50 > 10 nM T66665 CS4XN1 11994185 IC50 > 50000 nM T66665 C56TAE 11999248 IC50 = 130 nM T66665 CV29NY 12015271 IC50 = 6000 nM T66665 C4GP2H 12080914 IC50 > 100000 nM T66665 CA93XY 12088668 IC50 = 4000 nM T66665 CV32RZ 12088669 IC50 = 4000 nM T66665 CNE6W8 12088670 IC50 = 8 nM T66665 C4KJ0C 12266574 IC50 = 4688 nM T66665 CPKA02 12305221 IC50 > 40000 nM T66665 CJ65IL 12305517 IC50 > 40000 nM T66665 C0FX5O 12306155 IC50 > 40000 nM T66665 CKNP83 12309637 IC50 > 100000 nM T66665 C0X1AE 12310283 IC50 > 40000 nM T66665 CCZL29 12315005 IC50 > 10000 nM T66665 CZ87CS 12333000 IC50 = 94 nM T66665 CGQ2H9 12794430 IC50 = 7900 nM T66665 CELM69 12801541 IC50 > 40000 nM T66665 C6X9AH 12951906 IC50 = 75000 nM T66665 CVD83O 12965791 IC50 = 2 nM T66665 C7VR8X 12965792 IC50 = 0.14 nM T66665 CTB2Z6 12965793 IC50 = 0.36 nM T66665 C5TP0I 12990550 IC50 = 28000 nM T66665 C2K7BP 13125707 IC50 = 290 nM T66665 CQL7T8 13148385 IC50 = 22000 nM T66665 CUAN95 13148390 IC50 > 100000 nM T66665 C0SZJ2 13148391 IC50 > 100000 nM T66665 CTH23W 13148392 IC50 = 2000 nM T66665 CHM37E 13148394 IC50 = 12200 nM T66665 C5L7XU 13148395 IC50 = 2400 nM T66665 C0TOW4 13260662 IC50 = 81 nM T66665 C7HRX2 13260663 IC50 = 59 nM T66665 CPE4D9 13609513 IC50 > 100000 nM T66665 C6BR7D 13609518 IC50 > 100000 nM T66665 CST9K7 13771052 IC50 > 100000 nM T66665 CYK3G6 13804275 IC50 > 100000 nM T66665 CZQW71 13845711 IC50 = 15490 nM T66665 CM2NZ8 13986997 IC50 = 19400 nM T66665 CE0D3W 14015948 IC50 > 100000 nM T66665 C5EYL8 14049818 IC50 > 100000 nM T66665 C19KXV 14256046 IC50 = 5940 nM T66665 CV1WD7 14256049 IC50 = 2168 nM T66665 CC6S0G 14354678 IC50 = 500 nM T66665 CRB23M 14489592 IC50 = 41 nM T66665 CH7XB9 14762933 IC50 = 20 nM T66665 CS46EO 15153337 IC50 = 15 nM T66665 C4L7PE 15181201 IC50 > 40000 nM T66665 CD6A5Y 15192150 IC50 > 10000 nM T66665 CKQ06L 15293126 IC50 = 1096.48 nM T66665 CZ0FW1 15337398 IC50 = 0.02 nM T66665 CY43FD 15340372 IC50 = 70 nM T66665 C7KDB9 15345555 IC50 = 1318.26 nM T66665 C0MNT2 15345565 IC50 = 22 nM T66665 C9V0SW 15345568 IC50 = 12.88 nM T66665 CKB73V 15380222 IC50 > 100000 nM T66665 C7D5HB 15380227 IC50 > 100000 nM T66665 CXS52V 15388843 IC50 = 3000 nM T66665 CN4M6X 15388846 IC50 = 14 nM T66665 C1WVD9 15388847 IC50 = 3210 nM T66665 CIV0Q3 15390770 IC50 = 410 nM T66665 CR0QX1 15390771 IC50 = 10 nM T66665 CKOA87 15390773 IC50 = 2100 nM T66665 C7ZYU9 15406810 IC50 = 139.99 nM T66665 C20GFH 15428927 IC50 = 27 nM T66665 CFP7D1 15429218 IC50 = 270 nM T66665 C31OBS 15429221 IC50 = 18000 nM T66665 CFMC16 15429222 IC50 = 280 nM T66665 C1WDE7 15429226 IC50 = 1200 nM T66665 CI93RK 15431535 IC50 = 80 nM T66665 C0AFD5 15431540 IC50 = 20 nM T66665 C57CWU 15431541 IC50 = 40 nM T66665 CE81LY 15434168 IC50 = 670 nM T66665 CEK9A4 15453868 IC50 > 10000 nM T66665 C0F2NZ 15453869 IC50 = 6200 nM T66665 C90MOZ 15453870 IC50 = 2590 nM T66665 CB4R2G 15453871 IC50 = 570 nM T66665 CFZ3V5 15453872 IC50 = 170 nM T66665 CGQ15F 15453873 IC50 = 460 nM T66665 C9I4JX 15461522 IC50 > 10000 nM T66665 C6OVQ9 15461525 IC50 = 330 nM T66665 C8HE4A 15461526 IC50 = 1000 nM T66665 CUY31L 15461527 IC50 = 260 nM T66665 C1W8LT 15485017 IC50 = 540 nM T66665 CML5V6 15485782 IC50 = 24 nM T66665 CV0W5O 15485784 IC50 = 56 nM T66665 CRTS53 15485950 IC50 = 31000 nM T66665 C63KDN 15485951 IC50 > 300000 nM T66665 C1ZUI0 15516798 IC50 = 40 nM T66665 C3LIQ7 15516799 IC50 = 280 nM T66665 CT31VI 15516800 IC50 = 20 nM T66665 CYV58N 15521080 IC50 < 400 nM T66665 C8PEQ1 15521081 IC50 < 400 nM T66665 CC7J3Y 15524017 IC50 = 800 nM T66665 C5C4IJ 15551252 IC50 = 700 nM T66665 CY2O8J 15551254 IC50 = 50 nM T66665 C2BH3P 15600355 IC50 = 100 nM T66665 CYDT38 15617384 IC50 = 20 nM T66665 C72QCS 15871000 IC50 = 20 nM T66665 CTS5M8 15871001 IC50 = 3100 nM T66665 C6VK2B 15871995 IC50 = 33000 nM T66665 CUXL06 15871996 IC50 = 147000 nM T66665 CCB6R7 15871997 IC50 = 14000 nM T66665 C2MW9E 15871999 IC50 = 33000 nM T66665 C6LEP5 15887626 IC50 = 20 nM T66665 C2Z7BD 15887860 IC50 < 200 nM T66665 CY31HD 15887862 IC50 < 200 nM T66665 CTZN57 15887864 IC50 < 200 nM T66665 CHT0D5 15887866 IC50 < 200 nM T66665 CC09IL 15887878 IC50 < 200 nM T66665 C1S4MQ 16007065 IC50 = 1.8 nM T66665 CCJ15Y 16007066 IC50 = 1.9 nM T66665 C3D6ZR 16007330 IC50 = 360 nM T66665 C1SUI7 16036827 IC50 = 16040 nM T66665 CK94IN 16036828 IC50 = 18450 nM T66665 C89WYZ 16038368 IC50 > 100000 nM T66665 C2MH6N 16045730 IC50 > 10000 nM T66665 CNGD87 16072151 IC50 = 310 nM T66665 C9GNW0 16086577 IC50 > 10 ug.mL-1 T66665 CEJZ01 16098411 IC50 > 100000 nM T66665 C1XGO9 16098419 IC50 > 100000 nM T66665 CH4RY6 16125421 IC50 = 20000 nM T66665 C0KTX5 16125422 IC50 > 100000 nM T66665 CH8PR5 16125423 IC50 = 29000 nM T66665 C86XQV 16125424 IC50 = 16000 nM T66665 C4P3AM 16125427 IC50 = 56000 nM T66665 CHR83T 16125428 IC50 > 100000 nM T66665 C8HKG4 16125488 IC50 = 6900 nM T66665 C1PC2X 16125489 IC50 = 14000 nM T66665 CX5WF4 16125491 IC50 = 76000 nM T66665 C9TL4Z 16415139 IC50 > 100000 nM T66665 C0ZLK6 16605209 IC50 = 560 nM T66665 CE6J5R 16659826 IC50 = 42500 nM T66665 CHZ67I 16679964 IC50 > 33100 nM T66665 CMPG07 16679966 IC50 = 10100 nM T66665 C2DJ0O 16680045 IC50 = 6900 nM T66665 CU94BZ 16680046 IC50 > 34900 nM T66665 C03ETJ 16681478 IC50 = 90200 nM T66665 C4ZK0P 16730269 IC50 = 3000 nM T66665 CK96FW 16741227 IC50 = 100 nM T66665 CDA6Y0 16741228 IC50 = 280 nM T66665 CCPS15 16753427 IC50 > 10 nM T66665 C7M5CP 16753431 IC50 > 10 nM T66665 CS92DA 16753475 IC50 > 10 nM T66665 CN8WX3 16757526 IC50 = 1700 nM T66665 CHX45B 16774693 IC50 > 100000 nM T66665 CPY46E 16774950 IC50 > 100000 nM T66665 COL01E 16777326 IC50 > 100000 nM T66665 C98EUS 17128416 IC50 = 1400 nM T66665 CJHY01 17128417 IC50 = 4840 nM T66665 CH30KU 17128418 IC50 = 1560 nM T66665 CIO72R 17128419 IC50 = 1390 nM T66665 C6QIX5 17128427 IC50 = 2240 nM T66665 CZ71OR 17128430 IC50 = 1390 nM T66665 C15ULP 17128433 IC50 = 1210 nM T66665 CSH3B0 17128441 IC50 = 10590 nM T66665 C1U7OF 17128445 IC50 = 2700 nM T66665 COX86H 17128446 IC50 = 440 nM T66665 CKV16Q 17128476 IC50 = 930 nM T66665 C1ITN4 17128477 IC50 = 160 nM T66665 CVAD68 17128481 IC50 = 7400 nM T66665 CXPT85 17816126 IC50 = 610 nM T66665 C82XZE 17816357 IC50 = 29 nM T66665 C4NZB0 17828963 IC50 > 30000 nM T66665 C8VBA3 17876325 IC50 > 30000 nM T66665 CKX7R6 17876403 IC50 > 30000 nM T66665 C3IF4O 17880562 IC50 < 400 nM T66665 C52AKR 17919591 IC50 = 500 nM T66665 CB76TO 17919592 IC50 = 30 nM T66665 CZAV04 17919601 IC50 = 260 nM T66665 C5WHF9 17919602 IC50 = 50 nM T66665 CZ3Y4S 17919604 IC50 = 1300 nM T66665 CN78MC 17919609 IC50 = 1100 nM T66665 CNA75S 18400189 IC50 = 670 nM T66665 CME6G0 18400199 IC50 = 5100 nM T66665 CIB46D 18542198 IC50 = 39.6 nM T66665 C32YUX 18542229 IC50 = 15.7 nM T66665 COY2S1 18542237 IC50 = 6.77 nM T66665 CHW34K 18542252 IC50 = 128 nM T66665 CM29WC 18542265 IC50 = 41.5 nM T66665 CHN16W 18542282 IC50 = 421 nM T66665 CS8JB4 18542341 IC50 = 2200 nM T66665 CWD09Y 18542351 IC50 = 414 nM T66665 CR3MG9 18542368 IC50 = 5.68 nM T66665 C2KQ6W 18543182 IC50 > 100000 nM T66665 CTL49C 18678268 IC50 > 100000 nM T66665 C1Q0ZN 18701559 IC50 = 2100 nM T66665 CW4V5S 18933706 IC50 = 2 nM T66665 CC85QH 18946587 IC50 = 4300 nM T66665 CWF4D0 18969710 IC50 = 5 nM T66665 CBQL15 18969715 IC50 = 2.2 nM T66665 C2L4QT 18969738 IC50 = 110 nM T66665 CJ24BR 18969753 IC50 = 96 nM T66665 C9D4ZV 18969762 IC50 > 5000 nM T66665 C6U5AR 18969768 IC50 = 530 nM T66665 C8JHM7 18972826 IC50 = 12 nM T66665 C1U4YK 18972828 IC50 = 8 nM T66665 C0XP7E 18972838 IC50 = 14 nM T66665 CL19DP 18998922 IC50 = 190 nM T66665 C5U2ZR 19001581 IC50 = 6840 nM T66665 C9ZGX8 19361705 IC50 = 40 nM T66665 CP85SE 19426793 IC50 = 230 nM T66665 CNFL01 19594572 IC50 < 200 nM T66665 C46SER 19815165 IC50 = 55000 nM T66665 C89PVS 20055661 IC50 > 40000 nM T66665 CP34MI 20115449 IC50 > 100000 nM T66665 CP5EU3 20117519 IC50 > 100000 nM T66665 CX36PZ 20402500 IC50 = 19.32 nM T66665 CL0ZP4 20516107 IC50 = 210 nM T66665 C9V5YH 20516370 IC50 = 290 nM T66665 CTU20F 20658522 IC50 > 30000 nM T66665 CF7BY0 20658551 IC50 = 1600 nM T66665 CF93ID 20675009 IC50 > 50000 nM T66665 CGR8X6 20769058 IC50 > 40000 nM T66665 CLX62I 20826014 IC50 > 5000 nM T66665 C49YZM 20876816 IC50 = 407380.28 nM T66665 C7VLN6 21223973 IC50 = 87000 nM T66665 C2XRA6 21223977 IC50 = 57000 nM T66665 CRF1N2 21472741 IC50 = 380 nM T66665 CGP84X 21472742 IC50 = 800 nM T66665 CDJI26 21472746 IC50 = 250 nM T66665 CF9A1O 21472747 IC50 = 69 nM T66665 C8XH0M 21472750 IC50 = 500 nM T66665 C7SMC9 21472751 IC50 = 550 nM T66665 C19WHN 21472753 IC50 = 1200 nM T66665 C7D9QM 21472754 IC50 = 3200 nM T66665 C29VBS 21472759 IC50 = 200 nM T66665 C6U7PD 21545764 IC50 = 13450 nM T66665 C24QKO 21596130 IC50 = 46400 nM T66665 CK49UX 21626480 IC50 > 50000 nM T66665 CUSW63 21626481 IC50 > 50000 nM T66665 CX8CM6 21630094 IC50 > 50000 nM T66665 C8VR9H 21699911 IC50 = 5000 nM T66665 CZUT41 21837604 IC50 = 43 nM T66665 CBS0C1 21858549 IC50 > 5000 nM T66665 CGC46S 21859783 IC50 = 110 nM T66665 CA1GV2 21859784 IC50 = 120 nM T66665 C1QV5P 21859785 IC50 = 40 nM T66665 C0VW7T 21859786 IC50 = 30 nM T66665 C4CQN5 21862750 IC50 = 4140 nM T66665 CI14XS 21883501 IC50 = 73 nM T66665 C24DNQ 21883549 IC50 = 110 nM T66665 C97AWR 21883555 IC50 = 43 nM T66665 CO12EU 21883567 IC50 = 18 nM T66665 C60ZGU 21883595 IC50 = 250 nM T66665 COU74S 21883604 IC50 = 21.1 nM T66665 C3AQW5 21883607 IC50 = 21300 nM T66665 CRSU56 21883613 IC50 = 110 nM T66665 CNW0V1 21883621 IC50 = 100 nM T66665 CMY42K 21883631 IC50 = 140 nM T66665 CVG02E 21948438 IC50 = 90 nM T66665 C2FQO3 21948445 IC50 = 150 nM T66665 C0HEC8 21948463 IC50 = 350 nM T66665 CA09OG 21948479 IC50 = 1700 nM T66665 C41OLJ 21948498 IC50 = 30 nM T66665 C2KU0M 21948499 IC50 = 620 nM T66665 CF9E3P 21948521 IC50 = 40 nM T66665 CH7B4D 21948533 IC50 = 260 nM T66665 C9I8LB 22034354 IC50 = 470 nM T66665 CQ9WG2 22034355 IC50 > 40000 nM T66665 CYAS85 22034360 IC50 = 110 nM T66665 CLB58M 22034361 IC50 = 5900 nM T66665 CB2F0T 22034364 IC50 = 20 nM T66665 CH9E6Y 22034366 IC50 > 40000 nM T66665 CX6Q7U 22034367 IC50 = 300 nM T66665 CMV2E3 22034374 IC50 = 770 nM T66665 C3T6WH 22034376 IC50 = 110 nM T66665 CZ2UB6 22034379 IC50 = 570 nM T66665 CBDG24 22034386 IC50 = 1090 nM T66665 CF2N0H 22148957 IC50 = 5000 nM T66665 CVK2C0 22148978 IC50 = 1200 nM T66665 C30ZDS 22277772 IC50 = 70 nM T66665 CRGD86 22285759 IC50 = 85.1 nM T66665 C6O7NY 22285760 IC50 = 0.54 nM T66665 CYG05Q 22285769 IC50 = 3.133 nM T66665 CFW25L 22285770 IC50 = 5 nM T66665 C5O9LB 22285771 IC50 = 5.15 nM T66665 CYHT74 22285775 IC50 = 5 nM T66665 CJ80RW 22285776 IC50 = 0.7998 nM T66665 CT47ZF 22285778 IC50 = 0.2799 nM T66665 CRJ08O 22285779 IC50 = 0.3698 nM T66665 CKI4F5 22285780 IC50 = 1.41 nM T66665 CJW31Q 22285782 IC50 = 6.44 nM T66665 C2LRW6 22285784 IC50 = 0.02 nM T66665 C62QGV 22315630 IC50 = 3311.31 nM T66665 C08IZM 22562341 IC50 = 51 nM T66665 CWRA65 22624559 IC50 > 100000 nM T66665 CO2X7W 22643554 IC50 = 39.81 nM T66665 CF8M0T 22907695 IC50 = 27 nM T66665 CNL89X 22911749 IC50 = 110 nM T66665 CDOE75 22911767 IC50 = 350 nM T66665 CM6HA9 22911810 IC50 = 23 nM T66665 C3A4JD 22911832 IC50 = 270 nM T66665 CHY0X9 22911835 IC50 = 9 nM T66665 C3U6GI 22911939 IC50 > 30000 nM T66665 CFID36 22911970 IC50 = 2480 nM T66665 CX5IO1 22911977 IC50 = 13 nM T66665 CT9Y7O 22911990 IC50 = 57 nM T66665 CVOW97 22912028 IC50 = 18 nM T66665 CI0C2S 22912091 IC50 = 10 nM T66665 C9JP4B 22912100 IC50 = 7 nM T66665 C0XL3N 22912115 IC50 = 16 nM T66665 C0CT3B 22912123 IC50 = 1600 nM T66665 CBG45C 22912143 IC50 = 520 nM T66665 C8NS9E 22912151 IC50 = 32 nM T66665 CX5B4Y 22912186 IC50 = 21 nM T66665 CK4W3Z 22912196 IC50 = 430 nM T66665 C8GI4S 22912244 IC50 = 79 nM T66665 C54EBF 22912306 IC50 = 10 nM T66665 CW59QG 23002400 IC50 = 8800 nM T66665 CJYI21 23003613 IC50 = 9.81 nM T66665 CZV7D6 23225437 IC50 = 140 nM T66665 C4M8AQ 23356595 IC50 = 41000 nM T66665 CQ8O0J 23497471 IC50 = 272 nM T66665 CIJS71 23627031 IC50 > 100000 nM T66665 CC9PI3 23634884 IC50 = 2100 nM T66665 C62UXO 23663407 IC50 = 10100 nM T66665 CASU54 23696973 IC50 > 100000 nM T66665 C6UE8A 23717031 IC50 = 20000 nM T66665 CTQ9L0 24205505 IC50 = 2.1 nM T66665 C6DTY4 24689970 IC50 > 100000 nM T66665 CBR5L7 24695790 IC50 > 100000 nM T66665 CC8JB3 24721570 IC50 > 10000 nM T66665 CBU06J 24740875 IC50 = 50 nM T66665 COV92E 24752865 IC50 = 210000 nM T66665 CLV9T5 24816384 IC50 > 10 nM T66665 CELN62 24816405 IC50 = 1160 nM T66665 CD8PF6 24816406 IC50 = 640 nM T66665 C4B5MX 24824762 IC50 = 10600 nM T66665 CGS50Y 24825528 IC50 = 170 nM T66665 CSJ30T 24825529 IC50 = 270 nM T66665 COG2F3 24825530 IC50 = 250 nM T66665 C7O6GJ 24825531 IC50 = 1000 nM T66665 C4M2IO 24825532 IC50 = 440 nM T66665 C2FN0W 24825533 IC50 = 85 nM T66665 C5ZV1E 24825635 IC50 > 2000 nM T66665 CZFA18 24825636 IC50 = 2400 nM T66665 C03MQR 24825637 IC50 = 1000 nM T66665 CW1V6K 24825638 IC50 = 66000 nM T66665 C6H0GW 24825639 IC50 = 4000 nM T66665 CQ2P0C 24825640 IC50 = 1200 nM T66665 CHFJ48 24825641 IC50 = 300 nM T66665 C6Z3NL 24828801 IC50 > 10 nM T66665 C70QHI 24828802 IC50 > 10 nM T66665 CUNJ72 24848656 IC50 = 245470.89 nM T66665 C4QEA8 24850953 IC50 = 1290 nM T66665 C85UXM 24853947 IC50 > 100000 nM T66665 C57ERS 24853948 IC50 > 100000 nM T66665 CP0DT5 24853949 IC50 > 100000 nM T66665 CV3ZL6 24853950 IC50 > 100000 nM T66665 CZ91QG 24854030 IC50 > 100000 nM T66665 CO8FU7 24854031 IC50 > 100000 nM T66665 C83WEO 24854032 IC50 > 100000 nM T66665 CQ1Z3E 24867180 IC50 = 600 nM T66665 C4IP5C 24871714 IC50 = 8400 nM T66665 C57CPS 24882361 IC50 = 300006041.1 nM T66665 CE7TF2 24951013 IC50 = 1300 nM T66665 C2F9XY 24971276 IC50 > 10 nM T66665 C69YHL 25000755 IC50 = 47.2 nM T66665 CKP7C5 25044152 IC50 = 8000 nM T66665 C46WQB 25058950 IC50 = 9100 nM T66665 CB0E2M 25071014 IC50 = 11000 nM T66665 CWAR61 25072270 IC50 = 770 nM T66665 COMP96 25072271 IC50 = 730 nM T66665 CP9GS2 25116312 IC50 = 17510 nM T66665 CF0RV1 25116313 IC50 = 16340 nM T66665 CB5D9U 25116314 IC50 = 17500 nM T66665 CO5YQ2 25116315 IC50 = 16630 nM T66665 C24TUP 25116316 IC50 = 21010 nM T66665 C46WEF 25116556 IC50 = 20110 nM T66665 C1WQ7F 25141098 IC50 = 5700 nM T66665 CEFW12 25141402 IC50 = 3800 nM T66665 C6RZC2 25147690 IC50 > 10 nM T66665 C0PAE1 25179516 IC50 > 10 nM T66665 CWP75F 25179517 IC50 > 10 nM T66665 CM7I6Q 25179710 IC50 > 10 nM T66665 CG57UY 25179711 IC50 > 10 nM T66665 C5RBW3 25179712 IC50 > 10 nM T66665 CL3Q7B 25179713 IC50 > 10 nM T66665 C54DIT 25179907 IC50 > 40000 nM T66665 CTDF23 25179908 IC50 > 10 nM T66665 C9GB6J 25179909 IC50 > 10 nM T66665 C68FHV 25179910 IC50 > 10 nM T66665 CC9N3E 25179911 IC50 > 10 nM T66665 CUTK18 25179912 IC50 > 10 nM T66665 CAVM57 25187677 IC50 > 20000 nM T66665 C3Y1RA 25188731 IC50 < 1000 nM T66665 CN8VX0 25188732 IC50 = 3800 nM T66665 CU1BY0 25188733 IC50 = 3200 nM T66665 CY30US 25188735 IC50 = 3500 nM T66665 CPG9H1 25211353 IC50 = 2800 nM T66665 CHD71R 25242339 IC50 = 10200 nM T66665 C12DQW 25258347 IC50 = 190 nM T66665 CF92JB 25258348 IC50 = 730 nM T66665 C7H1IW 25258349 IC50 = 1820 nM T66665 CZ05XC 25258350 IC50 = 690 nM T66665 CJ3GP2 25261944 IC50 = 87 nM T66665 CMY91X 25768158 IC50 = 140 nM T66665 C1KA0H 25768159 IC50 = 240 nM T66665 CIY0W2 29335654 IC50 = 53 nM T66665 CB24VZ 30680185 IC50 = 2410 nM T66665 CKJ82C 38864639 IC50 = 54640 nM T66665 CF3WI1 39917259 IC50 = 11120 nM T66665 C7ADW8 40688876 IC50 = 13120 nM T66665 C8CWK5 42605184 IC50 = 31800 nM T66665 CXU63O 42607532 IC50 = 15000 nM T66665 CY19CJ 42609839 IC50 < 1000 nM T66665 C6DAY7 42609841 IC50 < 1000 nM T66665 CR7D1Q 43335949 IC50 > 50000 nM T66665 C8DQ4J 43358934 IC50 > 100000 nM T66665 C3SHI8 44138220 IC50 = 2500 nM T66665 C8DXK6 44143712 IC50 = 4330 nM T66665 C95VMW 44194809 IC50 = 270 nM T66665 CR0ZJ5 44194810 IC50 = 34000 nM T66665 CCI14S 44194811 IC50 = 68200 nM T66665 C4G7KU 44194812 IC50 > 100000 nM T66665 CE8B1R 44194813 IC50 = 17200 nM T66665 CJ8MZ9 44194814 IC50 > 100000 nM T66665 CCZ52W 44194816 IC50 > 100000 nM T66665 CP7F6J 44219621 IC50 = 1700 nM T66665 CF0JK5 44219631 IC50 = 6400 nM T66665 CF5A4V 44230565 IC50 = 2000 nM T66665 CIE70A 44250139 IC50 = 57 nM T66665 CR68BA 44250281 Ki > 25118.86 nM T66665 C8C7HF 44266438 IC50 > 33000 nM T66665 C7LT2W 44266451 IC50 = 21000 nM T66665 CC6W5I 44266508 IC50 = 18000 nM T66665 CGO38W 44269688 IC50 = 5000 nM T66665 C1W6AG 44271105 IC50 > 100000 nM T66665 CYHD60 44271141 IC50 > 100000 nM T66665 CP14AY 44271257 IC50 = 24 nM T66665 C1ZT4X 44271312 IC50 = 5 nM T66665 C0KMS2 44271350 IC50 = 59 nM T66665 CVC65J 44271374 IC50 = 28 nM T66665 C9Q7AY 44271388 IC50 = 18 nM T66665 CR18XW 44271618 IC50 = 140 nM T66665 C6HY3T 44271914 IC50 = 290 nM T66665 C3AQB6 44271916 IC50 = 100 nM T66665 CD0G2T 44271975 IC50 = 200 nM T66665 C65LRW 44271985 IC50 = 90 nM T66665 CPFB09 44272072 IC50 = 140 nM T66665 CT5JK3 44272073 IC50 = 7500 nM T66665 CAH19S 44272086 IC50 = 70 nM T66665 CW1V9M 44272115 IC50 = 1900 nM T66665 CR97YP 44272129 IC50 > 33000 nM T66665 CCG76A 44272130 IC50 > 33000 nM T66665 CA12DG 44272131 IC50 = 310 nM T66665 CVP23I 44272272 IC50 = 4300 nM T66665 C8M5HD 44272274 IC50 = 24000 nM T66665 C84VER 44272279 IC50 = 320 nM T66665 C62UAH 44272281 IC50 = 110 nM T66665 C59XIC 44272282 IC50 = 3200 nM T66665 CBPS42 44274898 IC50 = 47 nM T66665 CQG5R6 44274910 IC50 = 210 nM T66665 CY8QC3 44275200 IC50 = 110 nM T66665 C0MWO6 44275214 IC50 = 320 nM T66665 CCPX07 44275215 IC50 = 85 nM T66665 CJSE28 44275226 IC50 = 330 nM T66665 C8VK3W 44275248 IC50 = 220 nM T66665 C12ZHN 44275426 IC50 = 190 nM T66665 CBWA12 44275560 IC50 = 370 nM T66665 CSA4V0 44275675 IC50 = 110 nM T66665 CW8AY1 44275695 IC50 = 170 nM T66665 C5W4RT 44275714 IC50 = 500 nM T66665 C89LGZ 44275745 IC50 = 120 nM T66665 CWRF71 44275772 IC50 = 7 nM T66665 CGN3S5 44275809 IC50 = 7 nM T66665 CNH7D2 44275824 IC50 = 30 nM T66665 CMDE94 44275919 IC50 = 390 nM T66665 CTC2U6 44286188 IC50 = 30 nM T66665 C74AXR 44286194 IC50 = 1000 nM T66665 C3DQM8 44286210 IC50 = 360 nM T66665 C16ZON 44286326 IC50 = 49 nM T66665 C7HM5U 44286327 IC50 = 11000 nM T66665 C1I7BA 44286343 IC50 = 310 nM T66665 CYFP05 44286434 IC50 = 870 nM T66665 CZ8YW9 44286540 IC50 = 220 nM T66665 C0GH2Z 44286564 IC50 = 1700 nM T66665 CHC54N 44288984 IC50 = 7500 nM T66665 C0D8JY 44289750 IC50 = 850 nM T66665 CG7E9I 44290866 IC50 = 530 nM T66665 C39MAJ 44291228 IC50 = 230 nM T66665 CO7QL1 44291231 IC50 = 2900 nM T66665 C1LX6V 44291232 IC50 = 760 nM T66665 CD57LQ 44291249 IC50 = 2640 nM T66665 CK6CW2 44291335 IC50 = 770 nM T66665 C75LHO 44291336 IC50 = 265 nM T66665 CJA6R4 44291367 IC50 = 150 nM T66665 C47LVG 44291579 IC50 = 8000 nM T66665 C1VXS3 44291698 IC50 = 550 nM T66665 C4P2QA 44291754 IC50 = 129 nM T66665 C2PX9L 44292803 IC50 < 200 nM T66665 CQ8VR4 44292819 IC50 < 200 nM T66665 C5MCZ4 44292887 IC50 < 200 nM T66665 CPM5C9 44293185 IC50 < 200 nM T66665 CP16JH 44293186 IC50 < 200 nM T66665 CPS6C2 44293290 IC50 < 200 nM T66665 CNG5E2 44293477 IC50 = 1000 nM T66665 CN5FO1 44293478 IC50 = 980 nM T66665 CNJ6W7 44293738 IC50 = 1000 nM T66665 C40VHQ 44293755 IC50 = 280 nM T66665 CLJ6N1 44293775 IC50 = 220 nM T66665 C0BM5Q 44293785 IC50 = 1000 nM T66665 CF7J1T 44293786 IC50 = 300 nM T66665 CMG7L9 44293798 IC50 = 310 nM T66665 C7SYX6 44293966 IC50 = 340 nM T66665 CY4IZ3 44293967 IC50 = 950 nM T66665 C9GIL0 44293982 IC50 = 1200 nM T66665 CB5ZI8 44293983 IC50 = 1050 nM T66665 C6BQR4 44293986 IC50 = 280 nM T66665 CPH1M8 44294002 IC50 = 1050 nM T66665 CST64C 44294003 IC50 = 320 nM T66665 CHI4Y0 44295247 IC50 > 5000 nM T66665 C4YA8T 44307351 IC50 > 30000 nM T66665 CY4C8G 44307447 IC50 > 30000 nM T66665 CN2YL4 44307454 IC50 = 5400 nM T66665 C0TCY3 44307455 IC50 = 7200 nM T66665 C3Y1FP 44307489 IC50 = 550 nM T66665 CANV95 44307492 IC50 > 30000 nM T66665 CZ8QF9 44307510 IC50 > 30000 nM T66665 C7LH0E 44307511 IC50 > 30000 nM T66665 CBRU60 44307554 IC50 > 30000 nM T66665 CU80YE 44307569 IC50 > 100000 nM T66665 CAT54L 44307599 IC50 > 30000 nM T66665 CYK0M4 44307760 IC50 > 30000 nM T66665 CBSP93 44307761 IC50 > 30000 nM T66665 CU73YD 44309741 IC50 = 6870684.4 nM T66665 CAE0I2 44309745 IC50 = 835795.45 nM T66665 CQ2GW4 44309749 IC50 = 2236145.2 nM T66665 CEI94B 44309766 IC50 = 7048553.49 nM T66665 CVG78K 44309825 IC50 = 936052.05 nM T66665 CF5LB1 44309826 IC50 = 1425607.59 nM T66665 C1KT2G 44309833 IC50 = 1478427.39 nM T66665 CX6F7T 44309928 IC50 = 2343689.1 nM T66665 CZ8SQ6 44309929 IC50 = 720111.92 nM T66665 C5CD9I 44309952 IC50 = 1386117.35 nM T66665 CZ23EF 44310048 IC50 = 87902.25 nM T66665 CG2XF7 44310053 IC50 = 1416772.11 nM T66665 CFE19W 44310160 IC50 = 1760759.34 nM T66665 C2ZCE5 44310162 IC50 = 33000 nM T66665 C1IJ9A 44310164 IC50 = 6309573.44 nM T66665 CV93XP 44310188 IC50 = 1080936.05 nM T66665 CY6ML0 44310222 IC50 = 23000 nM T66665 C82SQB 44316044 IC50 = 93 nM T66665 CJ2A1Y 44316046 IC50 = 20 nM T66665 C9K2HM 44316112 IC50 = 100 nM T66665 CPUF05 44316113 IC50 = 7 nM T66665 CQVU84 44316126 IC50 = 11 nM T66665 CA9W4P 44316373 IC50 = 5 nM T66665 CS8P4H 44323766 IC50 > 30000 nM T66665 CLN5J2 44323818 IC50 > 33000 nM T66665 CP4V8T 44323830 IC50 > 100000 nM T66665 CZ0RT7 44323831 IC50 > 33000 nM T66665 CK93EF 44324030 IC50 = 12 nM T66665 CL36JK 44325870 IC50 = 3960 nM T66665 CAU4X9 44325888 IC50 = 1832 nM T66665 C2KB1O 44326499 IC50 = 610 nM T66665 CL6G5D 44326522 IC50 = 1330 nM T66665 CQ5HM8 44326892 IC50 = 16 nM T66665 C74TXM 44326894 IC50 = 3800 nM T66665 CCF6N9 44327823 IC50 = 39.81 nM T66665 CYH73O 44327824 IC50 = 75 nM T66665 CG95FW 44327825 IC50 = 32 nM T66665 CBK0Y9 44327826 IC50 = 6 nM T66665 C9XN8L 44327837 IC50 = 1500 nM T66665 CQF89I 44327838 IC50 = 16 nM T66665 C52FEI 44327839 IC50 = 9 nM T66665 CMHZ15 44327884 IC50 = 21 nM T66665 CUH0C2 44330273 IC50 > 300000 nM T66665 CL3E5I 44330326 IC50 = 19000 nM T66665 C19PLO 44330414 IC50 = 9 nM T66665 C9G4VJ 44330429 IC50 > 100000 nM T66665 C8K7MC 44330479 IC50 = 10000 nM T66665 CBY7I3 44330480 IC50 = 130000 nM T66665 C5LQJ9 44330483 IC50 > 300000 nM T66665 C7SU3C 44330495 IC50 = 66000 nM T66665 C0ZJ3M 44330496 IC50 = 49000 nM T66665 CO5RF2 44330530 IC50 = 200000 nM T66665 C2Z7VQ 44330531 IC50 > 300000 nM T66665 CBA30Q 44330561 IC50 = 6000 nM T66665 C6YV5C 44330563 IC50 = 101000 nM T66665 CYR60M 44330592 IC50 = 86000 nM T66665 CZD2L4 44330600 IC50 = 13000 nM T66665 CJ3CA1 44330646 IC50 = 30 nM T66665 CN0VW2 44336299 IC50 = 70 nM T66665 C74VEH 44336308 IC50 = 14 nM T66665 CSA3H6 44336320 IC50 > 100000 nM T66665 CB3Q2P 44336321 IC50 = 19000 nM T66665 C4C6QR 44336366 IC50 = 190 nM T66665 C78ANR 44338168 IC50 = 550 nM T66665 C0TNX5 44338327 IC50 = 40 nM T66665 C43QKL 44338544 IC50 = 30 nM T66665 CN6AS1 44338764 IC50 = 4168.69 nM T66665 CQVO89 44338793 IC50 = 524.81 nM T66665 C02TAU 44339126 IC50 = 83.18 nM T66665 CTIM78 44339284 IC50 = 169.82 nM T66665 CV07XW 44343489 IC50 = 6 nM T66665 C53XTU 44343803 IC50 = 2 nM T66665 C6IUT2 44343844 IC50 > 1000 nM T66665 CMKY74 44343870 IC50 = 274 nM T66665 C5H0EO 44343879 IC50 = 284 nM T66665 C4GM9U 44343958 IC50 > 1000 nM T66665 CR3F9L 44344532 IC50 = 35 nM T66665 CP6C3D 44344591 IC50 = 3000 nM T66665 C5OU6Q 44344842 IC50 = 15 nM T66665 C0QGP5 44344893 IC50 > 100000 nM T66665 CWKA30 44358995 IC50 = 2100 nM T66665 CD43ME 44363057 IC50 > 40000 nM T66665 CR04WS 44364343 IC50 = 1950 nM T66665 CUK06R 44364344 IC50 = 3300 nM T66665 CG7F5Q 44364345 IC50 = 6300 nM T66665 C7PFL4 44364510 IC50 = 51200 nM T66665 CGV0I9 44364554 IC50 = 1990 nM T66665 C3EWB8 44364555 IC50 = 712 nM T66665 CZN51K 44364565 IC50 = 7050 nM T66665 CE5P6X 44364615 IC50 = 5000 nM T66665 CI96RA 44364629 IC50 = 760 nM T66665 CU57KF 44364630 IC50 = 2800 nM T66665 CR38ZN 44364666 IC50 = 6850 nM T66665 CR5TP7 44364684 IC50 = 901 nM T66665 CGS1V5 44364699 IC50 = 1380 nM T66665 C9X0UY 44364814 IC50 = 28600 nM T66665 C2I4UH 44365341 IC50 = 3600 nM T66665 CN53LW 44365508 IC50 > 5000 nM T66665 CX64FE 44365531 IC50 > 5000 nM T66665 CA8RK2 44365569 IC50 > 5000 nM T66665 CBG3R5 44365570 IC50 = 1000 nM T66665 CJ7Z3V 44365691 IC50 = 6000 nM T66665 CQ8KJ3 44365712 IC50 = 33000 nM T66665 CQN69G 44365713 IC50 = 2600 nM T66665 CKM4L8 44365743 IC50 = 420 nM T66665 CSVX52 44365745 IC50 = 5000 nM T66665 CTWC52 44365758 IC50 = 900 nM T66665 CP8MK0 44365764 IC50 > 5000 nM T66665 CU8NA9 44365785 IC50 = 66000 nM T66665 CTZD86 44365815 IC50 = 4000 nM T66665 C72KCH 44365816 IC50 = 6300 nM T66665 C5HOZ1 44365843 IC50 = 11000 nM T66665 CVI60L 44365854 IC50 = 3000 nM T66665 C15KCX 44365956 IC50 = 2000 nM T66665 C9OZ5T 44365958 IC50 = 60 nM T66665 CG2N8Y 44366012 IC50 > 20000 nM T66665 CE50RI 44366112 IC50 > 33000 nM T66665 C67VZW 44366425 IC50 = 4000 nM T66665 CZB0K1 44366500 IC50 = 21000 nM T66665 C69TCB 44366535 IC50 = 1300 nM T66665 C26CIT 44366550 IC50 = 770 nM T66665 C3OM8C 44366551 IC50 = 19000 nM T66665 C8R1HW 44366732 IC50 = 980 nM T66665 CCX61K 44366749 IC50 = 1800 nM T66665 CSA5O9 44366768 IC50 = 2600 nM T66665 C2BSY4 44366835 IC50 = 5600 nM T66665 CF4I6P 44366839 IC50 = 9700 nM T66665 CAJ6R5 44366863 IC50 = 20000 nM T66665 CH84ZU 44366864 IC50 = 9700 nM T66665 CH35MX 44366879 IC50 = 5600 nM T66665 CU0P1T 44366883 IC50 = 5000 nM T66665 C93SAN 44366892 IC50 = 8400 nM T66665 CD8OI9 44366915 IC50 = 7100 nM T66665 CG9IE8 44370479 IC50 = 700 nM T66665 C43QVB 44370496 IC50 = 60 nM T66665 C6PQ8I 44370503 IC50 = 700 nM T66665 CJUC35 44370506 IC50 = 50 nM T66665 C8X3GE 44370516 IC50 = 350 nM T66665 CER97H 44370520 IC50 = 200 nM T66665 C1FZ8D 44370521 IC50 = 50 nM T66665 CER2T7 44370528 IC50 > 33000 nM T66665 C2KAB9 44370560 IC50 = 600 nM T66665 C61DTQ 44370597 IC50 = 640 nM T66665 C8U0HS 44370604 IC50 = 2100 nM T66665 CZI0B6 44370618 IC50 > 10000 nM T66665 CM72JP 44370626 IC50 = 10000 nM T66665 CG4RK8 44370627 IC50 > 10000 nM T66665 CW21SL 44370636 IC50 = 1560 nM T66665 CFA7R3 44370649 IC50 = 1240 nM T66665 CV62SH 44370724 IC50 > 10000 nM T66665 CP3C8D 44370735 IC50 > 5000 nM T66665 C1JL9O 44370742 IC50 = 2400 nM T66665 CH9XR0 44370744 IC50 = 300 nM T66665 C9JG2T 44370777 IC50 = 3 nM T66665 C7EBG2 44370786 IC50 = 110 nM T66665 C5M3UI 44370787 IC50 = 200 nM T66665 CFB0R4 44370791 IC50 = 370 nM T66665 C23EBS 44370949 IC50 = 1300 nM T66665 CO8F6L 44371320 IC50 = 450 nM T66665 CZ6NB9 44371399 IC50 = 150 nM T66665 CRKX10 44371400 IC50 = 79432823.47 nM T66665 CG2LE1 44371407 IC50 = 32 nM T66665 CNAY39 44371411 IC50 = 260 nM T66665 CB1VP9 44371422 IC50 = 3 nM T66665 CF9M7G 44371423 IC50 = 22 nM T66665 CU87HG 44371424 IC50 = 3 nM T66665 C4EH5S 44371430 IC50 = 13 nM T66665 C0GSH9 44371442 IC50 > 50000 nM T66665 CZY89I 44371457 IC50 = 10000 nM T66665 CV5CT2 44371478 IC50 = 48 nM T66665 CJ1B2O 44371479 IC50 = 36 nM T66665 C09UKQ 44371492 IC50 = 6 nM T66665 C58UDX 44371493 IC50 = 11 nM T66665 CL2SU4 44371522 IC50 = 15 nM T66665 CH4V8C 44372792 IC50 > 10000 nM T66665 CNBA18 44373038 IC50 = 2630 nM T66665 C5QH4B 44373252 IC50 > 10000 nM T66665 CM3JR7 44373310 IC50 = 2770 nM T66665 C98KAQ 44373311 IC50 > 10000 nM T66665 CT03QD 44373312 IC50 = 384000 nM T66665 C64XZB 44373323 IC50 > 10000 nM T66665 CGJ0M7 44373324 IC50 > 10000 nM T66665 C5UC8Z 44373338 IC50 = 1470 nM T66665 CSB9D6 44373350 IC50 = 2270 nM T66665 C2S9ZH 44373645 IC50 > 10000 nM T66665 CK2G0U 44373646 IC50 > 10000 nM T66665 CL85CK 44373654 IC50 = 6250 nM T66665 C2IY7Z 44374212 IC50 = 38000 nM T66665 CO0Q1M 44374403 IC50 = 140 nM T66665 CXMA02 44378192 IC50 < 100 nM T66665 C84GOY 44378193 IC50 > 10000 nM T66665 CH3J8M 44378194 IC50 > 10000 nM T66665 CG0L4N 44378225 IC50 < 100 nM T66665 CKI2Y8 44382878 IC50 > 30000 nM T66665 C18EVN 44382879 IC50 > 30000 nM T66665 C8TXC1 44383014 IC50 > 300000 nM T66665 CV14NG 44383162 IC50 = 30000 nM T66665 CD91OG 44383293 IC50 = 38000 nM T66665 C4USH1 44383428 IC50 = 44000 nM T66665 C1QJ0T 44383441 IC50 > 30000 nM T66665 CGH80T 44383449 IC50 > 300000 nM T66665 C18OMN 44383556 IC50 > 300000 nM T66665 CG6YA9 44383560 IC50 > 30000 nM T66665 CG89SY 44383610 IC50 = 5900 nM T66665 COHY08 44383630 IC50 = 30000 nM T66665 C7DT4Q 44383772 IC50 > 30000 nM T66665 C59OQY 44383922 IC50 > 10000 nM T66665 C8D4RP 44384088 IC50 > 10000 nM T66665 CN9L7S 44384322 IC50 = 48000 nM T66665 CJZC85 44384324 IC50 = 194000 nM T66665 C9ZM5A 44384325 IC50 = 254000 nM T66665 C7UCT0 44384330 IC50 > 300000 nM T66665 CSJ45Z 44384383 IC50 > 300000 nM T66665 CH40GX 44384384 IC50 > 300000 nM T66665 CQN19A 44384436 IC50 > 300000 nM T66665 C8M7RO 44387158 IC50 = 50 nM T66665 CA25XP 44388803 IC50 = 32000 nM T66665 CIOV43 44388811 IC50 = 2000 nM T66665 CAI5Z2 44388920 IC50 = 31600 nM T66665 C0Z8SH 44392359 IC50 = 3380.65 nM T66665 C9A4FM 44393815 IC50 = 660 nM T66665 CCDH14 44393845 IC50 = 200 nM T66665 CO2RG9 44393852 IC50 = 200 nM T66665 C37BAX 44393874 IC50 = 1090 nM T66665 CI9P5S 44393917 IC50 = 1210 nM T66665 C0FH8A 44393943 IC50 = 800 nM T66665 CZ8DS4 44393974 IC50 > 40000 nM T66665 CON98R 44394040 IC50 = 6.918 nM T66665 CJA59H 44394041 IC50 = 3.981 nM T66665 CL48WZ 44394042 IC50 > 40000 nM T66665 CPL8V0 44394061 IC50 = 12.02 nM T66665 C0RU8B 44394065 IC50 = 3.981 nM T66665 CW35JE 44394100 IC50 = 12.88 nM T66665 C80QPC 44394101 IC50 = 3.02 nM T66665 C5NWA9 44394120 IC50 = 14.13 nM T66665 C8D3SC 44394128 IC50 = 6.026 nM T66665 C0LO6A 44394134 IC50 = 3.02 nM T66665 CT8Z6E 44394150 IC50 = 22.91 nM T66665 C2UE8J 44394151 IC50 = 5.012 nM T66665 CXKW31 44394152 IC50 = 338.84 nM T66665 CAC41P 44394156 IC50 = 32.36 nM T66665 C6HW1A 44394175 IC50 = 7.943 nM T66665 CW6PL2 44394178 IC50 = 6.026 nM T66665 CI3W1R 44394196 IC50 = 1.995 nM T66665 C7VCZ4 44394200 IC50 = 20.89 nM T66665 CNUF49 44394201 IC50 = 239.88 nM T66665 CJ4NK9 44394204 IC50 = 12.88 nM T66665 CE0MN4 44394205 IC50 = 5.012 nM T66665 CB1AQ6 44394206 IC50 = 83.18 nM T66665 CLO09F 44394229 IC50 = 1.995 nM T66665 C4BZ6J 44394233 IC50 = 5.012 nM T66665 CK87TF 44394245 IC50 = 12.88 nM T66665 C8CV7Q 44394246 IC50 = 20.89 nM T66665 CR3HM1 44394264 IC50 = 3.981 nM T66665 C5IV7B 44394265 IC50 = 10 nM T66665 CD5K3W 44394272 IC50 = 12.88 nM T66665 CFG2V3 44394275 IC50 = 19.05 nM T66665 C8MQU2 44394285 IC50 = 338.84 nM T66665 CKFM85 44394286 IC50 = 64.57 nM T66665 CAH37E 44395024 IC50 = 48 nM T66665 CTWD42 44395063 IC50 = 24 nM T66665 CE1O8I 44395070 IC50 < 10 nM T66665 C6GB9N 44395090 IC50 = 388 nM T66665 C5IJZ0 44395098 IC50 = 17 nM T66665 CYRL43 44395118 IC50 = 43 nM T66665 CK1CQ3 44395128 IC50 = 26 nM T66665 CM1C6S 44395142 IC50 = 13 nM T66665 CA58EW 44395152 IC50 = 264 nM T66665 C8V1IN 44395167 IC50 < 31 nM T66665 C60XRQ 44395168 IC50 = 50 nM T66665 CR9B7F 44395179 IC50 = 34 nM T66665 CG1JZ6 44395210 IC50 = 39 nM T66665 CH8KP6 44395250 IC50 = 57 nM T66665 C74OSX 44400364 IC50 = 7000 nM T66665 C01AGZ 44400756 IC50 = 20.89 nM T66665 CA0DF6 44400773 IC50 = 32.36 nM T66665 C40DPU 44400775 IC50 = 6.026 nM T66665 C5CW4S 44400928 IC50 = 15.85 nM T66665 CW89YC 44402559 IC50 = 1700 nM T66665 C9SJ2N 44404327 IC50 = 2 nM T66665 C27RWY 44404395 IC50 = 8 nM T66665 CJE4F9 44409570 IC50 = 600 nM T66665 CAG4S6 44413121 IC50 = 200 nM T66665 C8GKC7 44413139 IC50 = 250 nM T66665 C2T5CE 44413148 IC50 = 670 nM T66665 CH87VZ 44415454 IC50 = 11070 nM T66665 C6L1HD 44415455 IC50 = 12370 nM T66665 CM37ED 44424015 IC50 < 1000 nM T66665 C6UM5Y 44424016 IC50 = 6500 nM T66665 C2E8DO 44424403 IC50 > 100000 nM T66665 C9IJ0D 44424406 IC50 = 30 nM T66665 C25SCZ 44429859 IC50 = 490000 nM T66665 C7K8UC 44431346 IC50 = 630 nM T66665 CYBP49 44434498 IC50 = 2200 nM T66665 C59WCO 44435729 IC50 = 1500 nM T66665 CUPI01 44443328 IC50 = 150 nM T66665 CC04HF 44443330 IC50 = 160 nM T66665 CY5BC2 44447992 IC50 = 100 nM T66665 C7UR1D 44447993 IC50 = 100 nM T66665 CE83YO 44451317 IC50 = 28 nM T66665 C67VZR 44451433 IC50 = 36000 nM T66665 C5U8SJ 44451448 IC50 = 327 nM T66665 CA2O1E 44451451 IC50 = 3000 nM T66665 CQH0O5 44451472 IC50 = 629 nM T66665 C70HRS 44451473 IC50 = 166 nM T66665 C9O2HQ 44456510 IC50 = 5.1 nM T66665 C4ZA2J 44456513 IC50 = 31.1 nM T66665 CHR8J5 44456515 IC50 > 10000 nM T66665 C4LJ1A 44456517 IC50 > 10000 nM T66665 CF3AR6 44456542 IC50 = 93.9 nM T66665 CLE24C 44456543 IC50 = 9.8 nM T66665 CK6ZQ4 44456545 IC50 = 1916461.06 nM T66665 CH4L0D 44456548 IC50 > 10000 nM T66665 C3V5BJ 44456558 IC50 = 3130 nM T66665 CRU0P2 44456559 IC50 = 3720 nM T66665 CJX30N 44456566 IC50 = 25.3 nM T66665 CAY32Z 44456567 IC50 = 5.4 nM T66665 C0G7YQ 44456587 IC50 = 68.8 nM T66665 CP9H4R 44456591 IC50 = 11.7 nM T66665 C8V5SN 44456592 IC50 = 454.5 nM T66665 C62QNU 44456593 IC50 = 32.9 nM T66665 C9QMH1 44456607 IC50 = 4280 nM T66665 CB3I1C 44456613 IC50 = 33.7 nM T66665 CDM86Z 44456615 IC50 = 22.4 nM T66665 CL0RE7 44456616 IC50 = 102.8 nM T66665 CE93JC 44456617 IC50 = 527.8 nM T66665 C03QCT 44456618 IC50 = 211.3 nM T66665 C6TQ9U 44456619 IC50 = 475.9 nM T66665 CL9M6O 44456620 IC50 = 238.5 nM T66665 CMB97J 44456621 IC50 = 7760 nM T66665 C4JI3D 44456622 IC50 > 10000 nM T66665 CH3BO6 44456631 IC50 = 5090 nM T66665 CL6X3Y 44456635 IC50 = 36.7 nM T66665 C0FVH3 44456638 IC50 > 10000 nM T66665 CQK4E3 44456639 IC50 = 44.4 nM T66665 CP8I3Y 44456640 IC50 = 635 nM T66665 C69WKN 44456641 IC50 > 10000 nM T66665 C0ZOP8 44456642 IC50 = 728.6 nM T66665 C05SXU 44456643 IC50 > 10000 nM T66665 CIHG87 44456655 IC50 = 6540 nM T66665 CH89VO 44456656 IC50 = 1950 nM T66665 CV4EJ0 44456662 IC50 = 120.9 nM T66665 C85HOA 44456663 IC50 = 459.7 nM T66665 CI54RU 44456664 IC50 = 28.8 nM T66665 CZR07A 44456665 IC50 = 712 nM T66665 CL1CO0 44456666 IC50 = 1480 nM T66665 CXB52E 44456684 IC50 = 38.2 nM T66665 C48PKJ 44456687 IC50 = 18 nM T66665 C2P8OL 44456688 IC50 > 10000 nM T66665 CR72TZ 44456689 IC50 = 272.3 nM T66665 CZ1H7U 44456690 IC50 > 10000 nM T66665 C16DSJ 44456691 IC50 > 10000 nM T66665 CK2A6G 44456693 IC50 = 5.92 nM T66665 C3JR8V 44456710 IC50 = 7.5 nM T66665 CGYW45 44456711 IC50 = 2.4 nM T66665 C78ZOH 44456712 IC50 > 10000 nM T66665 C27EMU 44456713 IC50 = 140 nM T66665 CSR28J 44456714 IC50 = 15.2 nM T66665 C8FTG4 44456715 IC50 = 298.5 nM T66665 CH41XD 44456716 IC50 = 14.4 nM T66665 C8VJF9 44456737 IC50 = 163938138.7 nM T66665 CUOB37 44456738 IC50 = 37.6 nM T66665 C7A8TQ 44456739 IC50 = 1920 nM T66665 CJA41U 44456740 IC50 = 300.3 nM T66665 CFWT53 44456741 IC50 = 1890 nM T66665 CE1SN9 44456742 IC50 > 10000 nM T66665 CRIE24 44456743 IC50 > 10000 nM T66665 CMFS70 44456763 IC50 = 9.2 nM T66665 CHZ8P6 44456766 IC50 = 10.3 nM T66665 C61CMH 44456767 IC50 > 10000 nM T66665 CEL5T8 44456768 IC50 = 273.8 nM T66665 CVR51B 44456769 IC50 > 10000 nM T66665 C1U0CR 44456770 IC50 = 3000 nM T66665 CD9XU5 44456771 IC50 > 10000 nM T66665 CI43GO 44456772 IC50 = 51.9 nM T66665 C8ASD0 44456773 IC50 = 46.5 nM T66665 C50GVY 44456798 IC50 = 1930 nM T66665 C6YL0O 44456799 IC50 = 5720 nM T66665 C67TDR 44456800 IC50 = 157.6 nM T66665 C96MQY 44456801 IC50 = 3330 nM T66665 CMQ0A6 44456822 IC50 = 144.5 nM T66665 C3H4GR 44456824 IC50 = 90.7 nM T66665 CTX63G 44456825 IC50 = 1.2 nM T66665 C0H6MQ 44456826 IC50 = 77.2 nM T66665 CEZ8P0 44456839 IC50 = 1.2 nM T66665 CL6Q1O 44456840 IC50 = 41494448.81 nM T66665 CFU78H 44456841 IC50 = 10.9 nM T66665 C1XA2D 44456842 IC50 = 48.4 nM T66665 C05DQN 44456860 IC50 = 3980 nM T66665 CT7HE1 44456861 IC50 = 1210 nM T66665 C3TDZ4 44456883 IC50 = 0.4 nM T66665 CY4W2F 44456885 IC50 = 4.1 nM T66665 C7ZHV1 44456887 IC50 > 10000 nM T66665 CLJ73Y 44456888 IC50 > 10000 nM T66665 C7BLA2 44456890 IC50 = 527.8 nM T66665 C2XWI4 44460175 IC50 > 100000 nM T66665 CS4J0Y 44473488 IC50 = 2560 nM T66665 CNW37Q 44473489 IC50 = 21900 nM T66665 CD0AT5 44473490 IC50 = 18600 nM T66665 CD30GC 44473491 IC50 = 12030 nM T66665 CZ4C8E 44473492 IC50 > 100000 nM T66665 C2A4KE 44473493 IC50 = 8150 nM T66665 CPN75T 44473494 IC50 > 100000 nM T66665 C0MK9H 44473495 IC50 = 10830 nM T66665 C1AIL9 44473650 IC50 = 3740 nM T66665 CUE30M 44473651 IC50 > 100000 nM T66665 C6J2RO 44473652 IC50 = 2440 nM T66665 CMV3R2 44473653 IC50 = 13530 nM T66665 CUW67Z 44474131 IC50 = 2110 nM T66665 CO92ZS 44474132 IC50 = 270 nM T66665 CB25PR 44474133 IC50 = 410 nM T66665 C0FX4E 44474277 IC50 = 120 nM T66665 CJ9GH7 44474278 IC50 = 910 nM T66665 CUPE26 44474279 IC50 = 2690 nM T66665 C4JO6Z 44474280 IC50 = 450 nM T66665 CCKA05 44474281 IC50 = 460 nM T66665 CS20YU 44474282 IC50 = 7240 nM T66665 CF34OX 44474283 IC50 = 240 nM T66665 C54TCU 44474284 IC50 = 910 nM T66665 C5W2HM 44475682 IC50 = 8810 nM T66665 C58AIG 44475683 IC50 > 100000 nM T66665 CSEV14 44475684 IC50 > 100000 nM T66665 C7LM9A 44475685 IC50 = 21610 nM T66665 CJG1Z8 44475687 IC50 = 330 nM T66665 C1MKA9 44475839 IC50 = 1620 nM T66665 CXZ6M4 44475840 IC50 = 2530 nM T66665 CN20QC 44475841 IC50 = 1580 nM T66665 C3KSY1 44475842 IC50 = 160 nM T66665 C2JL7C 44475844 IC50 = 9380 nM T66665 CFA7N0 44475845 IC50 = 730 nM T66665 C52LKE 44475846 IC50 = 5930 nM T66665 CBV2U8 44537892 IC50 = 900 nM T66665 C8RW9E 44537992 IC50 = 1800 nM T66665 C30XPZ 44541795 IC50 = 530 nM T66665 C35GON 44559963 IC50 > 100000 nM T66665 CM7N8F 44563734 IC50 = 16000 nM T66665 C18NSI 44563762 IC50 = 21300 nM T66665 CQ50LO 44563767 IC50 = 1570 nM T66665 CJE82G 44563770 IC50 = 2540 nM T66665 CY24ED 44563802 IC50 = 820 nM T66665 C04FCZ 44563805 IC50 = 470 nM T66665 CTB3C7 44563806 IC50 = 1780 nM T66665 CC71OE 44563807 IC50 = 12800 nM T66665 C61AIS 44563811 IC50 = 1740 nM T66665 C25APK 44563999 IC50 > 50000 nM T66665 C41VKB 44564000 IC50 > 50000 nM T66665 CUN32V 44564002 IC50 = 1100 nM T66665 C2AW1B 44564048 IC50 = 50000 nM T66665 COU62Y 44564506 IC50 > 50000 nM T66665 CAPI90 44564507 IC50 = 50000 nM T66665 CWBL04 44570751 IC50 = 9400 nM T66665 CWC38B 44570752 IC50 = 3700 nM T66665 C0UA4H 44570789 IC50 = 5100 nM T66665 CSDE13 44570790 IC50 = 6000 nM T66665 CRT8Q1 44571459 IC50 = 2200 nM T66665 C2A7RC 44571462 IC50 = 17700 nM T66665 CXZ1U2 44571463 IC50 = 3300 nM T66665 CDL15O 44571464 IC50 = 14800 nM T66665 CTPV42 44571509 IC50 = 1740 nM T66665 C27FZM 44573406 IC50 = 2700 nM T66665 CMH6D1 44574027 IC50 = 600 nM T66665 C20LVW 44574046 IC50 = 2200 nM T66665 CU28BQ 44574047 IC50 = 9300 nM T66665 CKT85S 44577800 IC50 = 1300 nM T66665 C3DU8S 44577801 IC50 = 14000 nM T66665 CB1E6X 44577804 IC50 = 13500 nM T66665 CXE3G5 44581926 IC50 = 150 nM T66665 C82KLY 44581927 IC50 = 2500 nM T66665 CN0RZ4 44581928 IC50 = 2500 nM T66665 C48XMK 44581929 IC50 > 10000 nM T66665 C41WAT 44581930 IC50 = 190 nM T66665 CN01BJ 44581931 IC50 = 210 nM T66665 CU9R8L 44581948 IC50 = 170 nM T66665 CGWQ85 44581949 IC50 = 360 nM T66665 CVA10P 44582812 IC50 = 25430 nM T66665 CA04YB 44582833 IC50 = 65720 nM T66665 CXB2G4 44583798 IC50 > 100000 nM T66665 CE8QI7 44584103 IC50 > 100 ug.mL-1 T66665 C5GOW9 44584170 IC50 = 19700 nM T66665 C8X9VH 44584274 IC50 = 400 nM T66665 C25YEN 44584287 IC50 = 180000 nM T66665 CB96SQ 44584307 IC50 = 120000 nM T66665 CWM9V2 44584310 IC50 = 600000 nM T66665 CZX97S 44586786 IC50 = 100 nM T66665 C0UT8E 44586787 IC50 = 10 nM T66665 CSX1H7 44586804 IC50 = 0.1799 nM T66665 CD2G5H 44587408 IC50 = 5800 nM T66665 CO28GQ 44587409 IC50 = 4560 nM T66665 C3WRM5 44587410 IC50 = 2700 nM T66665 C09XWJ 44587411 IC50 = 65000 nM T66665 CASI69 44587478 IC50 = 740 nM T66665 C1JKZ3 44587479 IC50 = 45000 nM T66665 CC0KB3 44590762 IC50 = 7000 nM T66665 CJ8QE5 44590815 IC50 = 5800 nM T66665 CN28MP 44590818 IC50 = 3400 nM T66665 CHU2N9 44593531 IC50 > 10 nM T66665 CX54EY 44818111 IC50 = 2000 nM T66665 CZ31PF 45267710 IC50 = 5 nM T66665 CV4YK9 45267715 IC50 = 16 nM T66665 C9MC8Z 45267716 IC50 = 1683 nM T66665 C9TV1Z 45267717 IC50 > 10000 nM T66665 C3WXL0 45267733 IC50 = 114 nM T66665 CUBH53 45267747 IC50 = 43 nM T66665 CNS9Z2 45267769 IC50 = 11 nM T66665 C1BRY0 45267770 IC50 = 7.2 nM T66665 CNW5D2 45268615 IC50 = 277 nM T66665 CD2K4X 45268625 IC50 = 56 nM T66665 CNP20Q 45268649 IC50 = 5.6 nM T66665 C2EUZ7 45269433 IC50 = 3 nM T66665 C2CBS0 45269451 IC50 < 10 nM T66665 CU46BW 45269475 IC50 > 7200 nM T66665 C9XER4 45269485 IC50 = 717 nM T66665 CHU45M 45269513 IC50 = 2.4 nM T66665 C2KAY8 45270280 IC50 > 10000 nM T66665 C09BLU 45270285 IC50 = 63 nM T66665 C8KT1R 45270290 IC50 < 10 nM T66665 C5KMT9 45270336 IC50 < 10 nM T66665 C8ETI0 45270348 IC50 = 1.3 nM T66665 CMY4J7 45270349 IC50 < 1.4 nM T66665 CI18ZS 45271088 IC50 = 29 nM T66665 CS07LK 45271115 IC50 < 10 nM T66665 C6NPR3 45271129 IC50 = 6323 nM T66665 CZU07P 45271135 IC50 = 12 nM T66665 CIR3V5 45271980 IC50 > 10000 nM T66665 C4BVM8 45271990 IC50 > 10000 nM T66665 CCBV52 45271997 IC50 = 33 nM T66665 CXTE06 45271998 IC50 < 10 nM T66665 C5AZ2N 45272015 IC50 = 45 nM T66665 C6D0RE 45272025 IC50 = 23 nM T66665 CLNJ85 45272026 IC50 = 5263 nM T66665 CY82CH 45272817 IC50 > 10000 nM T66665 C7RT6N 45272818 IC50 > 10000 nM T66665 CA6N3E 45272824 IC50 < 10 nM T66665 CMU54J 45272831 IC50 = 104 nM T66665 CR0FZ9 45272838 IC50 = 1135 nM T66665 C50WBE 45272855 IC50 = 686 nM T66665 CJO71V 45273765 IC50 > 10000 nM T66665 CI6TU8 45273784 IC50 = 1034 nM T66665 C0E4AV 45273799 IC50 > 4640 nM T66665 CZ6YD5 45273803 IC50 = 85 nM T66665 CF4C0H 45273829 IC50 = 5 nM T66665 CL6D9O 45484357 IC50 = 2300 nM T66665 C9D4QN 45484363 IC50 = 4600 nM T66665 CT1GZ5 45484364 IC50 = 3500 nM T66665 CTP6R9 45484365 IC50 = 900 nM T66665 CJ68NE 45487101 IC50 = 4400 nM T66665 CK5VY7 45487106 IC50 = 980 nM T66665 CXR73D 45487114 IC50 = 17600 nM T66665 CJ14YU 45487141 IC50 = 2600 nM T66665 CJX28F 46213934 IC50 > 10000 nM T66665 CWKS60 46216828 IC50 = 860 nM T66665 CGRF59 46216829 IC50 = 11100 nM T66665 CQRN43 46229713 IC50 = 17000 nM T66665 C15MXE 46230909 IC50 = 890 nM T66665 CL8X6A 46230910 IC50 = 2600 nM T66665 CI4CG5 46230911 IC50 = 1200 nM T66665 CDNF84 46230912 IC50 = 2400 nM T66665 C48QZA 46232823 IC50 = 15600 nM T66665 CCZE80 46232824 IC50 = 16800 nM T66665 C0S7EZ 46232873 IC50 = 12800 nM T66665 C3J8PA 46232874 IC50 = 7500 nM T66665 C6RV7G 46701878 IC50 > 10000 nM T66665 C26XVH 46830092 IC50 = 6400 nM T66665 CZMY40 46830339 IC50 = 1300 nM T66665 C6TWH7 46830360 IC50 = 5900 nM T66665 CV5ZO3 46837777 IC50 > 40000 nM T66665 CM3H5J 46837918 IC50 = 10900 nM T66665 CGI58K 46845031 IC50 = 53600 nM T66665 C9DRL8 46845033 IC50 = 197900 nM T66665 C48OCQ 46845035 IC50 = 109200 nM T66665 CRQ29W 46880352 IC50 > 50000 nM T66665 CN62CQ 46880353 IC50 > 100000 nM T66665 C3G5RE 46884417 IC50 = 8000 nM T66665 CY90RC 46884418 IC50 = 12900 nM T66665 C6AW1D 46884443 IC50 = 5500 nM T66665 CYPD43 46892801 IC50 > 400000 nM T66665 C8MXU2 46906688 IC50 = 87600 nM T66665 C68SVP 46906730 IC50 = 78300 nM T66665 CFL89P 46906732 IC50 = 101900 nM T66665 C0HYK2 46906734 IC50 = 126000 nM T66665 CZ1BI2 46906736 IC50 = 357200 nM T66665 CDY1P0 46906738 IC50 = 100000 nM T66665 CT39AY 46906740 IC50 = 85400 nM T66665 CAT0M6 46926545 IC50 < 28 nM T66665 C2PL3G 46927848 IC50 > 10000 nM T66665 CTF94K 46934113 IC50 = 1500 nM T66665 CQV64T 46934114 IC50 = 4700 nM T66665 CY49EO 46934115 IC50 = 6500 nM T66665 C51LXR 46934255 IC50 > 100000 nM T66665 C8SO3Z 46934256 IC50 = 25000 nM T66665 CA20ZG 46934257 IC50 > 100000 nM T66665 CFAR39 46934258 IC50 = 310 nM T66665 CZ1X6V 46934874 IC50 = 1200 nM T66665 CI8P0A 46937277 IC50 > 1000000 nM T66665 CYL16R 49765093 IC50 > 100000 nM T66665 CBF20G 49788596 IC50 = 370 nM T66665 CP03KU 49799224 IC50 = 6700 nM T66665 C0A2SK 49799225 IC50 = 6100 nM T66665 CV0SD4 49799226 IC50 = 7800 nM T66665 C9JL4Z 49799227 IC50 = 7900 nM T66665 CWYT40 49799228 IC50 = 7200 nM T66665 C8IP0B 49799229 IC50 = 8900 nM T66665 C1RA6K 49799230 IC50 = 7600 nM T66665 CU40RO 49799231 IC50 = 8800 nM T66665 CNR7J1 49799265 IC50 = 9000 nM T66665 CS4D9W 49799266 IC50 = 8500 nM T66665 CMS46L 49799267 IC50 = 6700 nM T66665 CBNJ36 49799268 IC50 > 50000 nM T66665 CZ28MX 49799269 IC50 > 50000 nM T66665 CBWS90 49799270 IC50 > 50000 nM T66665 C9L3UH 49799271 IC50 > 50000 nM T66665 CJQ4I0 49799272 IC50 > 50000 nM T66665 C0S2VP 49799273 IC50 > 50000 nM T66665 C78XZV 49804917 IC50 = 8400 nM T66665 CEHY29 49804918 IC50 = 13000 nM T66665 C6IWU7 49804919 IC50 = 35300 nM T66665 C8W3GR 49804920 IC50 > 100000 nM T66665 CQO37H 49805049 IC50 = 34400 nM T66665 CQD83P 49805050 IC50 > 100000 nM T66665 CC51BP 49805051 IC50 > 100000 nM T66665 C5L4CW 49805052 IC50 > 100000 nM T66665 C8JVU3 49805053 IC50 > 100000 nM T66665 C8XY3D 49805054 IC50 > 100000 nM T66665 C5MDK8 49805055 IC50 = 61600 nM T66665 C51KQC 49805174 IC50 > 100000 nM T66665 C8CER6 49805175 IC50 = 5000 nM T66665 C1LGX6 49805176 IC50 > 100000 nM T66665 C0HTK6 49805177 IC50 > 100000 nM T66665 CX6K0C 49805178 IC50 = 22000 nM T66665 C0S4FY 49805179 IC50 = 5100 nM T66665 CD8J0L 49805180 IC50 > 100000 nM T66665 CBK9A7 49805302 IC50 > 100000 nM T66665 CVD4T1 49805303 IC50 = 36300 nM T66665 CU34WJ 49805304 IC50 > 100000 nM T66665 CVI2E6 49805305 IC50 > 100000 nM T66665 CRV4K9 49805306 IC50 > 100000 nM T66665 CLR02I 49805307 IC50 = 92000 nM T66665 CM8EC7 49826588 IC50 = 2470 nM T66665 CG7EJ4 49837500 IC50 = 65000 nM T66665 C6V8JC 49845477 IC50 = 20000 nM T66665 CW39TN 49862884 IC50 = 1600 nM T66665 CU16QR 49862898 IC50 = 3900 nM T66665 C67UXI 49862899 IC50 = 14400 nM T66665 C8ZD6G 49862900 IC50 = 3300 nM T66665 CM07SN 49864393 IC50 = 11800 nM T66665 CIS62C 49864409 IC50 = 10700 nM T66665 C7BHR5 49864410 IC50 = 7700 nM T66665 CTD40I 49864411 IC50 = 22300 nM T66665 C2QCH8 49864438 IC50 > 100000 nM T66665 CZ9UD6 50901657 IC50 > 100000 nM T66665 C81CPJ 50906262 IC50 = 21700 nM T66665 C5LNY7 50906263 IC50 = 19630 nM T66665 CT0G8A 50906264 IC50 = 6770 nM T66665 CUWJ62 50906265 IC50 = 19830 nM T66665 C7T6OY 50906266 IC50 = 7610 nM T66665 CC1U5M 50906267 IC50 = 3200 nM T66665 C01HYS 50906487 IC50 = 50310 nM T66665 CT74BU 50906488 IC50 = 9350 nM T66665 C0K5TQ 50906490 IC50 = 31850 nM T66665 C4M2NP 50908173 IC50 = 940 nM T66665 CUK21S 50908400 IC50 = 470 nM T66665 CNHJ51 50908401 IC50 = 380 nM T66665 C7AL4X 51003554 IC50 = 13400 nM T66665 C03UJK 51003555 IC50 = 66 nM T66665 COX20E 51003556 IC50 = 339 nM T66665 C69NBQ 51039210 IC50 = 420 nM T66665 CFX39I 51039215 IC50 = 2300 nM T66665 CQM21U 51039216 IC50 = 15800 nM T66665 C9LV0J 51039217 IC50 = 630 nM T66665 CU7ST1 51346826 IC50 > 100000 nM T66665 C3M5DB 51346951 IC50 = 2000 nM T66665 CI85WG 51346952 IC50 = 45000 nM T66665 CT8HO6 51346953 IC50 = 2700 nM T66665 CB7WE5 51351150 IC50 > 100000 nM T66665 CK31TX 51360478 IC50 > 5000 nM T66665 C3UX7A 51360480 IC50 > 5000 nM T66665 C5FZC7 51360481 IC50 > 5000 nM T66665 CMG36K 52826130 IC50 = 420 nM T66665 CL6VB4 52826143 IC50 = 370 nM T66665 CF6X5T 52826146 IC50 = 460 nM T66665 CCG7T3 52918139 IC50 = 17640 nM T66665 C17IAT 52918154 IC50 = 8870 nM T66665 CSBE15 52918155 IC50 = 10350 nM T66665 C4Y9MC 52918156 IC50 = 15350 nM T66665 C78YAE 52936776 IC50 = 11100 nM T66665 C26WPM 52941067 IC50 = 48000 nM T66665 C1OEI4 52941415 IC50 = 43 nM T66665 C0FQK2 52941574 IC50 > 100000 nM T66665 CW5U1X 52941672 IC50 = 8500 nM T66665 CT4D1X 52942295 IC50 = 12200 nM T66665 CJFR43 52942521 IC50 = 758 nM T66665 CR47KD 52942604 IC50 = 16 nM T66665 CV27HX 52942642 IC50 = 680 nM T66665 C9OED7 52942694 IC50 = 100000 nM T66665 C2Y5DB 52942695 IC50 = 14 nM T66665 CZNJ67 52942809 IC50 = 31000 nM T66665 C0XOH5 52943192 IC50 = 3330 nM T66665 CZC8Q3 52943858 IC50 = 42 nM T66665 CK52YW 52944376 IC50 = 30 nM T66665 CI5BF1 52946122 IC50 > 100000 nM T66665 CM6CJ2 52946158 IC50 = 18600 nM T66665 CQ5X9F 52946285 IC50 = 1700 nM T66665 C4K6BH 52946883 Ki > 100000 nM T66665 CBM7U1 52946890 IC50 = 210 nM T66665 CZCN58 52948356 IC50 = 3100 nM T66665 CQD5M1 52948912 IC50 = 100000 nM T66665 C0TXV9 52949921 IC50 = 330 nM T66665 CI9BQ4 52950184 IC50 = 34000 nM T66665 C6DF9H 52951272 IC50 = 2000 nM T66665 C6VWE2 52951275 IC50 = 1000 nM T66665 CD8SA7 52951485 IC50 > 10000 nM T66665 CH1T5N 52951486 IC50 > 10000 nM T66665 CPU67E 52951487 IC50 > 10000 nM T66665 CBN86G 52951488 IC50 = 7000 nM T66665 CYZ4C6 52951489 IC50 > 10000 nM T66665 C51QFH 52951612 IC50 = 2500 nM T66665 CRH4E8 52951613 IC50 = 1000 nM T66665 CPTE73 52951614 IC50 > 10000 nM T66665 C9HUZ2 52951734 IC50 = 3000 nM T66665 C96TVC 52951735 IC50 = 700 nM T66665 CLN12R 52951736 IC50 = 2800 nM T66665 C7GFM3 52951862 IC50 > 10000 nM T66665 CFJQ74 52951863 IC50 > 10000 nM T66665 CUSD82 52951864 IC50 = 7000 nM T66665 CP6M1R 52951865 IC50 = 2000 nM T66665 CD32FZ 52951866 IC50 = 6000 nM T66665 CU51RA 52951990 IC50 = 1300 nM T66665 CDT5Z6 52951991 IC50 = 900 nM T66665 C3UEM7 53248884 IC50 = 11000 nM T66665 C1SA2Z 53249089 IC50 > 400000 nM T66665 C58DMR 53252516 IC50 > 10000 nM T66665 C6KTX4 53307430 IC50 = 2400 nM T66665 C06YVC 53316515 IC50 > 100000 nM T66665 CKD6L2 53316516 IC50 > 100000 nM T66665 C3EUV0 53316645 IC50 = 70 nM T66665 C61HIM 53316646 IC50 = 5 nM T66665 C1OJ0M 53316888 IC50 > 100000 nM T66665 CG79XF 53316889 IC50 > 100000 nM T66665 C26NMZ 53317589 IC50 = 150 nM T66665 CKT7G2 53317947 IC50 = 85 nM T66665 CEC68I 53318243 IC50 = 110000 nM T66665 CYJT73 53318566 IC50 = 21250 nM T66665 CK6NI5 53318567 IC50 = 25420 nM T66665 CQ0Z3T 53319059 IC50 = 21300 nM T66665 C50LRC 53319285 IC50 = 150 nM T66665 CA6H8Q 53319286 IC50 = 1980 nM T66665 CRM4A0 53319287 IC50 = 62200 nM T66665 C3AD1U 53319288 IC50 = 8 nM T66665 CTL23B 53320186 IC50 = 100000 nM T66665 CRIX73 53320474 IC50 = 40100 nM T66665 CG68TH 53320588 IC50 = 94 nM T66665 C2TO9G 53320589 IC50 < 28 nM T66665 CYJ7F1 53320590 IC50 = 1130 nM T66665 CL9R7F 53320894 IC50 = 200000 nM T66665 CX2WV0 53321196 IC50 = 13540 nM T66665 C6EO8G 53321885 IC50 = 340 nM T66665 CVB21L 53321886 IC50 = 870 nM T66665 CUTF34 53322523 IC50 = 19700 nM T66665 CE14JM 53322743 IC50 = 1820 nM T66665 CA2W6X 53322834 IC50 = 46 nM T66665 C0GAC7 53323100 IC50 = 6380 nM T66665 CVUN53 53323101 IC50 = 103 nM T66665 CUF68R 53323225 IC50 > 100000 nM T66665 CKL68J 53323226 IC50 = 96000 nM T66665 CY36BC 53323227 IC50 = 7 nM T66665 CLI0R1 53323460 IC50 = 736037.6 nM T66665 CM4L0D 53323860 IC50 = 18010 nM T66665 CQ5UV6 53324322 IC50 = 530 nM T66665 CFTY39 53324454 IC50 = 78.4 nM T66665 CJK86T 53324575 IC50 = 19 nM T66665 CHX7F1 53324576 IC50 = 1480 nM T66665 C9NE3C 53324577 IC50 = 140 nM T66665 CXHQ58 53324578 IC50 = 68 nM T66665 CN86CK 53325524 IC50 = 4640 nM T66665 CL37DN 53325623 IC50 = 43410 nM T66665 C68WVL 53325872 IC50 = 100000 nM T66665 C7HSA5 53325873 IC50 = 910 nM T66665 CZ70LU 53326920 IC50 = 28800 nM T66665 CY3OX0 53363314 IC50 > 10000 nM T66665 CB89CZ 53484143 IC50 = 43300 nM T66665 C4U5IX 53493001 IC50 = 27000 nM T66665 C12QTA 53733023 IC50 = 3000 nM T66665 CZJY42 54669869 IC50 = 3200 nM T66665 C6UAZ5 54669874 IC50 = 1700 nM T66665 CU9W8M 54680181 IC50 > 10000 nM T66665 C2IB5H 54682566 IC50 >= 30000 nM T66665 COZ9N1 54685766 IC50 > 100 ug.mL-1 T66665 CEK6X8 54686705 IC50 = 830 nM T66665 C4O1PT 54698884 IC50 = 510 nM T66665 C87GPY 54728405 IC50 > 68000 nM T66665 C0X6ZQ 54728406 IC50 = 33700 nM T66665 CC1Y9K 54728407 IC50 = 70000 nM T66665 CROP60 54728408 IC50 > 100000 nM T66665 C76ETO 54728409 IC50 = 95600 nM T66665 CR0E7X 54728410 IC50 = 95300 nM T66665 C1ZR3C 54728411 IC50 = 74700 nM T66665 CAP19Z 54728413 IC50 = 92600 nM T66665 C3IXM4 54728414 IC50 = 263000 nM T66665 C0NTK4 54728415 IC50 = 44400 nM T66665 CT3PE0 54728416 IC50 > 74800 nM T66665 CPD72H 54728417 IC50 = 94700 nM T66665 CFT90G 54728419 IC50 = 33700 nM T66665 C3XW4R 54728423 IC50 > 100000 nM T66665 C7DY8K 54728424 IC50 > 100000 nM T66665 C14MSR 54728428 IC50 > 100000 nM T66665 CG9ZC5 54728429 IC50 > 57700 nM T66665 C5GRB6 54754354 IC50 > 10000 nM T66665 C3YM2E 54754518 IC50 > 10000 nM T66665 C6R9ES 54764159 IC50 = 800 nM T66665 C79DVG 56589615 IC50 > 10000 nM T66665 CGC8D1 56598067 IC50 = 270 nM T66665 CXV96Y 56598068 IC50 = 500 nM T66665 C9LUN0 56599285 IC50 = 12210 nM T66665 CTHQ38 56599737 IC50 = 17670 nM T66665 CN3F5O 56641761 IC50 > 10000 nM T66665 C7ZI3H 56642018 IC50 > 10000 nM T66665 CU1G5A 56642290 IC50 > 10000 nM T66665 C0SM7Z 56642536 IC50 > 10000 nM T66665 C6TLW3 56642537 IC50 > 10000 nM T66665 C75TMQ 56643482 IC50 = 13000 nM T66665 C4RC3Y 56661768 IC50 = 23000 nM T66665 C1MIO4 56665210 IC50 = 290000 nM T66665 CU2HX5 56665212 IC50 = 420000 nM T66665 CJMI28 56665214 IC50 > 1000000 nM T66665 CX30HR 56665216 IC50 = 70000 nM T66665 C5QZK1 56668661 IC50 > 1000000 nM T66665 CHC69U 56668662 IC50 = 2000 nM T66665 CHS43U 56668663 IC50 = 540000 nM T66665 CFI7A8 56668664 IC50 = 49000 nM T66665 CS79OK 56668666 IC50 > 1000000 nM T66665 C9QLO1 56668668 IC50 = 36000 nM T66665 C60GOL 56668670 IC50 = 540000 nM T66665 CPY6S5 56668671 IC50 = 17000 nM T66665 C7JEP3 56672143 IC50 = 150000 nM T66665 CCW0G2 56672144 IC50 = 36000 nM T66665 CM3X4L 56672145 IC50 = 76000 nM T66665 CHX16S 56675533 IC50 = 72000 nM T66665 C23DNE 56675535 IC50 = 430000 nM T66665 CI48HR 56680050 IC50 = 4200 nM T66665 CE74XR 56682184 IC50 > 1000000 nM T66665 CI7AU6 56682186 IC50 = 20000 nM T66665 CV89NW 56924661 IC50 = 380 nM T66665 CT2SY4 56924662 IC50 = 0.2 nM T66665 CPQ2W0 56924668 IC50 = 4600 nM T66665 CRB5G2 56929489 IC50 = 1700 nM T66665 CS1J6W 56929588 IC50 = 640 nM T66665 CU6QX9 56929591 IC50 = 400 nM T66665 CTUE06 56931531 IC50 = 13550 nM T66665 CL16UQ 56949326 IC50 < 10000 nM T66665 CWXR01 56951565 IC50 = 7500 nM T66665 CLO87D 56964583 IC50 > 100000 nM T66665 CKL87T 56987559 IC50 = 48 nM T66665 C6IE9W 57345498 IC50 = 6000 nM T66665 C3I9HG 57345509 IC50 = 710 nM T66665 C2KS6Y 57345510 IC50 = 840 nM T66665 CR35DN 57345511 IC50 = 430 nM T66665 CG1PE6 57345517 IC50 = 320 nM T66665 CK2VP4 57345687 IC50 = 7000 nM T66665 C17XJW 57384031 IC50 = 85000 nM T66665 CABU73 57384032 IC50 = 15000 nM T66665 CYR45H 57384033 IC50 = 14000 nM T66665 C2ET0L 57390204 IC50 = 25600 nM T66665 CB6O5D 57390392 IC50 > 100000 nM T66665 C4O3HY 57391146 IC50 = 3400 nM T66665 CJCD09 57391147 IC50 = 1900 nM T66665 CV0NB5 57391368 IC50 = 6530 nM T66665 CQVU96 57391399 IC50 > 1000000 nM T66665 CEGM35 57391400 IC50 = 450000 nM T66665 CMKF47 57391410 IC50 = 140000 nM T66665 C21FWN 57392194 IC50 = 56000 nM T66665 CX5CY1 57392459 IC50 = 60 nM T66665 CC2AF6 57392917 IC50 = 6600 nM T66665 C27JKX 57392918 IC50 = 2800 nM T66665 CU4OY7 57392919 IC50 = 12100 nM T66665 C5RP6B 57392920 IC50 = 6300 nM T66665 CLR62X 57393171 IC50 = 450000 nM T66665 CV7PA3 57393176 IC50 = 110000 nM T66665 C76TYD 57393522 IC50 > 400000 nM T66665 CA72OL 57393840 IC50 = 2300 nM T66665 C7CN0I 57393841 IC50 = 1800 nM T66665 CS52FT 57393844 IC50 = 730 nM T66665 CAXT47 57393845 IC50 = 2990 nM T66665 CGBD79 57393943 IC50 > 100000 nM T66665 CBYQ62 57393944 IC50 > 100000 nM T66665 CMLU74 57393945 IC50 > 100000 nM T66665 CXI23L 57394660 IC50 = 3700 nM T66665 CPW0Y9 57394866 IC50 = 17500 nM T66665 C6WH3Z 57394899 IC50 = 200000 nM T66665 C26MQU 57395427 IC50 = 52600 nM T66665 CAQ1V7 57395579 IC50 = 1700 nM T66665 C1CDN4 57395676 IC50 = 15000 nM T66665 C2P6NT 57396409 IC50 = 8500 nM T66665 CM5J7X 57396410 IC50 = 2600 nM T66665 CWAI02 57396427 IC50 = 598 nM T66665 CN9YM3 57397474 IC50 > 100000 nM T66665 CU01IE 57398427 IC50 = 700000 nM T66665 COKJ32 57399158 IC50 = 62000 nM T66665 CN6Q1M 57399159 IC50 > 100000 nM T66665 C0ZMF5 57399160 IC50 = 87000 nM T66665 CY3JD8 57399161 IC50 = 32000 nM T66665 C2GJQ6 57399859 IC50 = 11700 nM T66665 CSEF30 57399860 IC50 = 5600 nM T66665 CP3X1J 57400089 IC50 = 350000 nM T66665 CKA2C4 57400090 IC50 = 500000 nM T66665 C5LH3V 57400903 IC50 = 15000 nM T66665 CV1K0D 57401637 IC50 = 4900 nM T66665 C2LK4N 57401638 IC50 = 7800 nM T66665 CZV54H 57401639 IC50 = 3600 nM T66665 C0VB8K 57401640 IC50 = 5600 nM T66665 CM0YK9 57401647 IC50 = 30.7 nM T66665 CT39LO 57401870 IC50 = 12400 nM T66665 CWIT56 57401898 IC50 > 1000000 nM T66665 CE82VR 57401899 IC50 = 180000 nM T66665 CU6W9N 57402570 IC50 = 880 nM T66665 CH29UE 57402675 IC50 = 69000 nM T66665 C20JKE 57403365 IC50 = 7900 nM T66665 CXCJ10 57403366 IC50 = 12600 nM T66665 C96XSV 57403614 IC50 = 21000 nM T66665 C8J5WL 57780764 IC50 > 100000 nM T66665 CJK1Y2 57780765 IC50 > 100000 nM T66665 CXY02N 57780766 IC50 > 100000 nM T66665 CWXK91 57780767 IC50 > 100000 nM T66665 C37LRH 57780770 IC50 > 100000 nM T66665 CBUG72 57780771 IC50 = 20440 nM T66665 C9JQL6 57780772 IC50 > 100000 nM T66665 CEYZ93 57780773 IC50 = 1100 nM T66665 C02TNX 57780777 IC50 > 100000 nM T66665 CK0RX3 57780779 IC50 > 100000 nM T66665 CHT38U 58661838 IC50 > 10000 nM T66665 C21WOV 58934890 IC50 = 28 nM T66665 CYLF64 59052441 IC50 = 190 nM T66665 C6D5TJ 60150646 IC50 = 4600 nM T66665 CSB7D5 60150647 IC50 = 2100 nM T66665 C4P7YV 60150648 IC50 = 2200 nM T66665 C5K6SY 60150649 IC50 = 10800 nM T66665 CXLV30 60155351 IC50 = 24100 nM T66665 CP5O0C 60155353 IC50 = 26300 nM T66665 CG68SH 60155450 IC50 = 14000 nM T66665 CS4Q0U 60155529 IC50 = 21300 nM T66665 CEU8V0 60155531 IC50 = 4100 nM T66665 CGQ15M 60155532 IC50 = 13000 nM T66665 CLX65R 60155533 IC50 = 4000 nM T66665 CY1B9U 60155534 IC50 = 8300 nM T66665 CL71GR 60163969 IC50 = 9880 nM T66665 CKT2M9 66554463 IC50 = 14 nM T66665 CP05UZ 66554464 IC50 = 400 nM T66665 CWQ0A9 66561560 IC50 > 5000 nM T66665 C97DBL 66695948 IC50 = 1400 nM T66665 CING95 67288784 IC50 = 2100 nM T66665 CA7F0J 68819643 IC50 = 1270 nM T66665 CH8WL2 70438810 IC50 = 98.03 nM T66665 CKB8T3 70681274 IC50 > 100000 nM T66665 C5VIW7 70682749 IC50 = 45500 nM T66665 C7GAV8 70682750 IC50 = 37800 nM T66665 C64QAN 70683360 IC50 = 6100 nM T66665 CRQ93O 70684829 IC50 = 24500 nM T66665 C0OJZ5 70684830 IC50 = 14400 nM T66665 CTH34G 70685460 IC50 = 6000 nM T66665 C6IB1N 70685640 IC50 = 910 nM T66665 C13DNZ 70687598 IC50 = 14700 nM T66665 C8WF9U 70687599 IC50 > 100000 nM T66665 CCHQ37 70687603 IC50 = 5500 nM T66665 C1JT5Z 70687604 IC50 > 100000 nM T66665 C4J6WZ 70687793 IC50 = 920 nM T66665 CWX6K9 70689055 IC50 = 51800 nM T66665 C71ADP 70689056 IC50 = 121700 nM T66665 CER8H3 70689656 IC50 = 21300 nM T66665 CJ6KR1 70689657 IC50 > 100000 nM T66665 CAU73D 70689835 IC50 > 5000 nM T66665 CVF2T0 70691164 IC50 = 63000 nM T66665 CF9Z0J 70691338 IC50 = 1580 nM T66665 CO5R3M 70691800 IC50 = 9200 nM T66665 CZN89O 70691989 IC50 > 5000 nM T66665 C7GA0D 70693277 IC50 = 45400 nM T66665 CQ5MI9 70693858 IC50 = 10900 nM T66665 CX21IT 70693859 IC50 = 39600 nM T66665 C4FPG1 70693860 IC50 > 100000 nM T66665 CI7V9Q 70694020 IC50 = 910 nM T66665 CS3DX0 70695366 IC50 = 78200 nM T66665 C03ZOD 70695367 IC50 = 20000 nM T66665 CM9I7E 70695562 IC50 = 270 nM T66665 CVH05L 70695977 IC50 > 100000 nM T66665 CYWT28 70696152 IC50 = 930 nM T66665 C2AX0N 71449035 IC50 = 500 nM T66665 C6JV8C 71449165 IC50 = 1800 nM T66665 CLTX08 71449872 IC50 > 100000 nM T66665 CYF7V6 71449873 IC50 > 100000 nM T66665 CQNY45 71449874 IC50 > 100000 nM T66665 CPER64 71451367 IC50 = 38710 nM T66665 CC8FT0 71451368 IC50 = 52390 nM T66665 C5US7V 71451683 IC50 > 100000 nM T66665 CNMJ64 71451684 IC50 > 100000 nM T66665 CG6P1S 71451685 IC50 = 2500 nM T66665 C8P9IM 71451686 IC50 > 100000 nM T66665 C0B2CS 71452803 IC50 = 1700 nM T66665 C8TNO2 71453171 IC50 = 8250 nM T66665 C0O7WF 71453172 IC50 = 1020 nM T66665 CML95K 71453515 IC50 = 46500 nM T66665 C2P0NY 71453516 IC50 > 100000 nM T66665 C1XVD0 71453517 IC50 > 100000 nM T66665 CSE3I6 71453518 IC50 > 100000 nM T66665 C2MYH8 71453519 IC50 > 100000 nM T66665 CLGT46 71454915 IC50 = 69940 nM T66665 CO2FN6 71455230 IC50 > 100000 nM T66665 CJV50T 71455799 IC50 = 10000 nM T66665 CY21GU 71457021 IC50 > 100000 nM T66665 C5OEK7 71457022 IC50 = 27800 nM T66665 C7RS5E 71457023 IC50 > 100000 nM T66665 CLC0O1 71457024 IC50 > 100000 nM T66665 CVG1Y6 71457025 IC50 > 100000 nM T66665 CF2PX3 71457026 IC50 > 100000 nM T66665 CEK51Y 71457577 IC50 = 12800 nM T66665 C0ME4D 71458538 IC50 = 16830 nM T66665 CC0K5A 71458539 IC50 = 12640 nM T66665 C4K8EF 71458879 IC50 > 100000 nM T66665 C5RKA8 71458880 IC50 > 100000 nM T66665 C0DKS5 71458881 IC50 > 100000 nM T66665 C4AXT8 71458882 IC50 > 100000 nM T66665 CZQ37B 71458883 IC50 > 100000 nM T66665 C7OW6J 71458884 IC50 > 100000 nM T66665 CIPV26 71460384 IC50 = 13190 nM T66665 C60GCV 71460385 IC50 = 50250 nM T66665 C1RO4M 71460691 IC50 > 100000 nM T66665 CDP53O 71460692 IC50 > 100000 nM T66665 C31CTR 71460693 IC50 > 100000 nM T66665 CS0KB2 71460694 IC50 > 100000 nM T66665 CCM28N 71460695 IC50 = 72300 nM T66665 COZ76P 71461641 IC50 = 570 nM T66665 CKPQ80 71462077 IC50 = 74910 nM T66665 CN29UJ 71462079 IC50 = 8430 nM T66665 CWC86O 71462406 IC50 > 100000 nM T66665 CAZ71T 71495779 IC50 = 8920 nM T66665 C5YVD4 71495780 IC50 = 9670 nM T66665 CC0F9V 71495781 IC50 = 5090 nM T66665 C3WYB9 71495782 IC50 = 12360 nM T66665 CO5N4Y 71495783 IC50 = 6750 nM T66665 CK3VM2 71495784 IC50 = 1020 nM T66665 C8JQ0X 71495885 IC50 = 8990 nM T66665 C5L3NI 71495887 IC50 = 1270 nM T66665 CBTR23 71495888 IC50 = 1360 nM T66665 CYEG63 71495889 IC50 = 9080 nM T66665 CQ3T6J 71495988 IC50 = 2010 nM T66665 CXSL48 71495989 IC50 = 4560 nM T66665 C2T8MR 71495990 IC50 = 12960 nM T66665 C90OJI 71495991 IC50 = 4670 nM T66665 CUT0L5 71495992 IC50 = 8060 nM T66665 C82AZY 71495993 IC50 = 10080 nM T66665 C5TN2R 71509482 IC50 > 10000 nM T66665 CI35CO 71509483 IC50 = 61 nM T66665 CL36SU 71509484 IC50 = 54 nM T66665 C3HKW2 71509485 IC50 = 43 nM T66665 C3QXF6 71509486 IC50 = 59 nM T66665 C1EHY3 71509487 IC50 = 39 nM T66665 C78ZJW 71509612 IC50 = 150 nM T66665 CL0NU3 71509613 IC50 = 63 nM T66665 CXN9L6 71509614 IC50 = 84 nM T66665 C3CGO8 71517057 IC50 = 670 nM T66665 CMP36Q 71517058 IC50 = 6800 nM T66665 C6MH2C 71517059 IC50 = 21200 nM T66665 CC5Y2Q 71517060 IC50 = 590 nM T66665 CU1HJ4 71517061 IC50 = 1800 nM T66665 CTJ07U 71517062 IC50 = 9800 nM T66665 CYJ59C 71517206 IC50 = 9200 nM T66665 C9Y2HC 71517208 IC50 = 7200 nM T66665 CCK24M 71517362 IC50 = 1100 nM T66665 C97MUN 71517363 IC50 = 3900 nM T66665 C9YCI3 71520910 IC50 = 1010 nM T66665 CPF2G8 71521123 IC50 = 1260 nM T66665 CFV62N 71521225 IC50 = 84.7 nM T66665 CEJU20 71521226 IC50 = 618 nM T66665 C2H8SM 71521227 IC50 = 296 nM T66665 C7XMC2 71583324 IC50 = 60 nM T66665 CX18FE 71583325 IC50 = 70 nM T66665 COLY35 71583326 IC50 = 100 nM T66665 CUCE37 71583327 IC50 = 280 nM T66665 C5H2JA 71583438 IC50 = 280 nM T66665 CWRF17 71583439 IC50 = 310 nM T66665 C2OAB4 71583440 IC50 = 50 nM T66665 CCL43F 71583441 IC50 = 80 nM T66665 CB91XC 71583442 IC50 = 110 nM T66665 CK37YJ 71583443 IC50 = 240 nM T66665 C1PH5V 71583444 IC50 = 310 nM T66665 C7T4GM 71583556 IC50 = 320 nM T66665 C8UA7K 71619203 IC50 > 50000 nM T66665 CK1BH2 71652197 IC50 = 6890 nM T66665 C6IFQ2 71652198 IC50 = 20090 nM T66665 CV6K8P 71652199 IC50 = 11120 nM T66665 CV4NQ3 71652200 IC50 = 15090 nM T66665 CVU9N1 71652201 IC50 = 6660 nM T66665 CA1I3B 71652364 IC50 = 12980 nM T66665 C3XR0J 71652365 IC50 = 6840 nM T66665 CPA68L 71652366 IC50 = 16430 nM T66665 C8E1DW 71652367 IC50 = 9080 nM T66665 CT4RC7 71652368 IC50 = 8010 nM T66665 CVU84Z 71652369 IC50 = 23160 nM T66665 CXVN32 71652528 IC50 = 6690 nM T66665 CY0Q2M 71652529 IC50 = 7090 nM T66665 CTQ6H0 71652530 IC50 = 10280 nM T66665 CT7Z9H 71652531 IC50 = 1980 nM T66665 C5MX2K 71652532 IC50 = 10280 nM T66665 CKY25V 71652533 IC50 = 1450 nM T66665 CYG5R6 71652683 IC50 = 8570 nM T66665 C8RI2F 71652684 IC50 = 5780 nM T66665 C7AYD3 71652685 IC50 = 1880 nM T66665 CEB1P0 71652686 IC50 = 8010 nM T66665 C52OGW 71652687 IC50 = 8870 nM T66665 CM6AU2 71655553 IC50 = 150 nM T66665 CPY76V 71682135 IC50 > 100000 nM T66665 CN3O0S 71682136 IC50 > 100000 nM T66665 CQG9Z8 71714062 IC50 = 14800 nM T66665 C2WM6B 71714209 IC50 = 1300 nM T66665 CLS75K 71716000 IC50 > 33000 nM T66665 CYL26P 71718474 IC50 > 33000 nM T66665 CWC7Y9 71720245 IC50 > 33000 nM T66665 C58PBX 71720415 IC50 = 934 nM T66665 CWQ9R4 71723168 IC50 = 1300 nM T66665 CG1KW4 71723169 IC50 = 6500 nM T66665 CTF9N0 71723170 IC50 = 1500 nM T66665 C3GZ2F 71723171 IC50 = 28000 nM T66665 CF6O3R 71723307 IC50 = 1200 nM T66665 C0CL5Z 71723308 IC50 = 13000 nM T66665 C8I3DQ 71723309 IC50 = 1100 nM T66665 CVMK69 71723310 IC50 = 1000 nM T66665 CT65QH 71723311 IC50 = 170 nM T66665 CPUV68 71723312 IC50 = 3400 nM T66665 CRSI34 71723313 IC50 = 27000 nM T66665 CM86GD 72722785 IC50 = 2500 nM T66665 CW16PM 72792469 IC50 = 430 nM T66665 C6K2ND 72945107 IC50 = 7900 nM T66665 COEA64 72945305 IC50 = 7300 nM T66665 CNVA83 73053907 IC50 = 69 nM T66665 C5RK7T 73054179 IC50 = 38 nM T66665 C3UIZ2 73054542 IC50 > 100000 nM T66665 CT3CR0 73054543 IC50 > 100000 nM T66665 C7TK2A 73054544 IC50 > 100000 nM T66665 CLF0Z2 73054545 IC50 > 100000 nM T66665 CO12YG 73054546 IC50 = 10800 nM T66665 C10GHA 73054547 IC50 > 100000 nM T66665 C42QSB 73054548 IC50 > 100000 nM T66665 C6W7BM 73054804 IC50 = 6200 nM T66665 C08ETJ 73054805 IC50 > 100000 nM T66665 C6MYR7 73054806 IC50 = 160 nM T66665 C60QWG 73054807 IC50 = 320 nM T66665 CGXB89 73054808 IC50 = 28800 nM T66665 CREM98 73054809 IC50 > 100000 nM T66665 C2WSN9 73054810 IC50 = 240 nM T66665 C8KVH2 73055091 IC50 > 100000 nM T66665 CH5MU3 73055092 IC50 = 170 nM T66665 CO1U2Z 73055093 IC50 > 100000 nM T66665 CLMV21 73333200 IC50 = 21000 nM T66665 CBTQ18 73333399 IC50 = 13700 nM T66665 C3MF2U 73335400 IC50 > 10000 nM T66665 C3QEG6 73335403 IC50 > 10000 nM T66665 CE25BK 73335501 IC50 > 10000 nM T66665 CZ90QC 73335502 IC50 > 10000 nM T66665 CZP84O 73335598 IC50 > 10000 nM T66665 CJ3BK2 73335600 IC50 > 10000 nM T66665 C06IFC 73335691 IC50 > 10000 nM T66665 CC4DW1 73335692 IC50 > 10000 nM T66665 C9JS7Z 73335693 IC50 > 10000 nM T66665 C43EUZ 73335785 IC50 > 10000 nM T66665 CU6MN9 73350378 IC50 > 50000 nM T66665 CXKH51 73356534 IC50 = 17300 nM T66665 CG4Z2K 75166651 IC50 = 2500 nM T66665 C2AE0Z 76309082 IC50 > 100000 nM T66665 C1GQO6 76309083 IC50 = 320 nM T66665 C8L4GN 76310082 IC50 = 6200 nM T66665 C1GJ6D 76310083 IC50 = 700 nM T66665 CWY14K 76310400 IC50 = 35090 nM T66665 CL1PM5 76310401 IC50 = 550 nM T66665 CYN6O9 76310402 IC50 = 2270 nM T66665 CZ4J8T 76310403 IC50 > 100000 nM T66665 C32DPL 76310435 IC50 = 9110 nM T66665 C8ZCA6 76311083 IC50 = 35000 nM T66665 C8G1HR 76311084 IC50 = 26000 nM T66665 CFQB07 76311577 IC50 = 32.9 nM T66665 CUFQ45 76312769 IC50 = 150 nM T66665 CNBQ86 76312770 IC50 = 5300 nM T66665 CT1B6E 76312771 IC50 = 1770 nM T66665 CG1QT2 76312772 IC50 = 2500 nM T66665 CC26KV 76312773 IC50 > 100000 nM T66665 C9MAL6 76313613 IC50 = 2700 nM T66665 C7B5UG 76314063 IC50 > 100000 nM T66665 C71MXA 76314064 IC50 = 1040 nM T66665 C9LWE3 76315140 IC50 = 1210 nM T66665 C29LXT 76316303 IC50 > 100000 nM T66665 CN71DA 76316304 IC50 = 2100 nM T66665 CJTO94 76316305 IC50 = 320 nM T66665 C8PY6T 76317113 IC50 = 5600 nM T66665 CN3IY0 76317622 IC50 = 36230 nM T66665 CW75NC 76317623 IC50 = 56760 nM T66665 C6LPX0 76317624 IC50 = 30740 nM T66665 CR0TN5 76317625 IC50 = 1960 nM T66665 CA7T1F 76317626 IC50 = 90 nM T66665 CY38AN 76317627 IC50 = 1570 nM T66665 CED02X 76317628 IC50 = 10050 nM T66665 CT4CI2 76319998 IC50 = 310 nM T66665 C2RAE9 76319999 IC50 = 3600 nM T66665 C9UG0J 76320000 IC50 = 32000 nM T66665 CE9U8A 76320001 IC50 = 110 nM T66665 CWUV56 76320831 IC50 = 2780 nM T66665 CX80WZ 76320832 IC50 = 3600 nM T66665 CS6M5L 76323663 IC50 = 320 nM T66665 CE7X9B 76323664 IC50 = 120 nM T66665 CJ3X1B 76326065 IC50 = 3980 nM T66665 C50VPI 76327239 IC50 = 280 nM T66665 CVOL05 76327240 IC50 > 100000 nM T66665 C4L2HX 76327241 IC50 = 32 nM T66665 CDF46T 76327242 IC50 = 33100 nM T66665 C8AYK0 76328049 IC50 = 3100 nM T66665 CC7O9K 76328514 IC50 = 300 nM T66665 C8DQT1 76328515 IC50 = 300 nM T66665 CX9LH5 76328516 IC50 = 20680 nM T66665 CGS82O 76329158 IC50 = 340 nM T66665 CVZ4K0 76330897 IC50 = 2000 nM T66665 CYZ8X6 76330898 IC50 = 630 nM T66665 CX1YG3 76330899 IC50 = 3300 nM T66665 C2HF7T 76330900 IC50 = 114 nM T66665 C5IME3 76332195 IC50 = 260 nM T66665 CNPC96 76332196 IC50 = 240 nM T66665 C3IA4X 76332818 IC50 = 460 nM T66665 CG5Q1T 76334476 IC50 = 7900 nM T66665 C47GNU 76334477 IC50 = 320 nM T66665 C9ILC1 76334478 IC50 = 970 nM T66665 C1O6XT 76334479 IC50 = 1000 nM T66665 CF17OX 76335317 IC50 = 2400 nM T66665 CL3W1Z 76335832 IC50 > 100000 nM T66665 CRTL25 77461108 IC50 = 5880 nM T66665 CQU7B2 77461109 IC50 = 3170 nM T66665 C6TEQ2 77461110 IC50 = 2950 nM T66665 C2R4HM 77461111 IC50 = 4760 nM T66665 C2FI7T 77461112 IC50 = 4340 nM T66665 CCY52O 77461113 IC50 = 2930 nM T66665 C1JQ9D 77461114 IC50 = 3880 nM T66665 CJ06VH 77461119 IC50 = 6 nM T66665 CWJ4N9 77461129 IC50 = 150 nM T66665 C7KSB4 78091888 IC50 = 190 nM T66665 C1GU3V 78091940 IC50 = 69 nM T66665 CS2V0C 86294758 IC50 = 6100 nM T66665 CZ1UA3 86294759 IC50 = 4200 nM T66665 CL8YU9 86294760 IC50 = 8600 nM T66665 CXB76I 86294761 IC50 = 8100 nM T66665 C0DV5U 86302470 IC50 = 670 nM T66665 C4O6TA 86302472 IC50 = 1340 nM T66665 C8CF5A 88749792 IC50 = 69820 nM T66665 C17WBJ 90035911 IC50 > 100000 nM T66665 CMBR21 90036150 IC50 > 100000 nM T66665 CG5BN7 90036171 IC50 > 100000 nM T66665 C18JIM 90036424 IC50 = 2700 nM T66665 C8BP2Q 90036448 IC50 > 100000 nM T66665 CMV52R 90036800 IC50 = 74300 nM T66665 CV0M4P 90036900 IC50 > 100000 nM T66665 CF05NR 90643435 IC50 = 500 nM T66665 CRU63T 90643436 IC50 = 1200 nM T66665 CLOF59 90643437 IC50 = 2300 nM T66665 C0GD5E 90643438 IC50 = 4400 nM T66665 CN7EX4 90643439 IC50 = 5500 nM T66665 CX91YZ 90643440 IC50 = 8700 nM T66665 CKM72W 90643441 IC50 = 38000 nM T66665 CI1E6X 90643442 IC50 = 39000 nM T66665 C76YKC 90643443 IC50 = 42000 nM T66665 CI9D7M 90643444 IC50 = 50000 nM T66665 CVJB81 90643445 IC50 = 53000 nM T66665 C19SKL 90643446 IC50 = 58000 nM T66665 CW2A6R 90643447 IC50 = 67000 nM T66665 CE7N2Q 90643681 IC50 = 2400 nM T66665 C5DLR2 90643682 IC50 = 4350 nM T66665 CO10ZA 90643683 IC50 = 3850 nM T66665 CRFN68 90643684 IC50 = 3500 nM T66665 CQR2T6 90643685 IC50 = 3980 nM T66665 C73HBN 90643686 IC50 = 5030 nM T66665 CS97HW 90643687 IC50 = 2300 nM T66665 CIF45T 90643688 IC50 = 4630 nM T66665 C26ZQJ 90643689 IC50 = 1900 nM T66665 CVTB83 90643690 IC50 = 3530 nM T66665 C9X7IS 90643691 IC50 = 2800 nM T66665 COR58K 90643692 IC50 = 5210 nM T66665 CFO91K 90643693 IC50 = 4680 nM T66665 CLD39A 90643694 IC50 = 2750 nM T66665 CT0BL2 90643695 IC50 = 9580 nM T66665 CDBK93 90643696 IC50 = 9870 nM T66665 CF2KN9 90643697 IC50 = 6420 nM T66665 CX1YR5 90643698 IC50 = 3800 nM T66665 CSI21P 90644329 IC50 > 10000 nM T66665 C7N8YE 90644330 IC50 > 10000 nM T66665 C0Q2XP 90644331 IC50 > 10000 nM T66665 CDX79W 90644332 IC50 > 10000 nM T66665 C07VSO 90644333 IC50 > 10000 nM T66665 CEF51J 90644334 IC50 > 10000 nM T66665 CBXH26 90644335 IC50 > 10000 nM T66665 C9EO0N 90644336 IC50 > 10000 nM T66665 CQG56R 90644337 IC50 > 10000 nM T66665 CTVJ69 90645106 IC50 = 17410 nM T66665 CYW8G5 90645107 IC50 = 11210 nM T66665 C1R6LU 90645108 IC50 = 27650 nM T66665 C5U8JA 90645109 IC50 = 38210 nM T66665 C8CKM6 90645110 IC50 > 100000 nM T66665 CYN86M 90645111 IC50 = 31450 nM T66665 C3EAW0 90645112 IC50 = 14760 nM T66665 C4XF1V 90645113 IC50 = 19320 nM T66665 C30WLJ 90645114 IC50 > 100000 nM T66665 CG6YO8 90645115 IC50 = 13320 nM T66665 CJZ4X5 90645116 IC50 > 100000 nM T66665 CF4EB2 90645121 IC50 = 15000 nM T66665 CB2E7N 90645122 IC50 > 100000 nM T66665 CR2VS4 90645123 IC50 = 14850 nM T66665 C1ZYO3 90645124 IC50 = 27960 nM T66665 CYG4D2 90645131 IC50 = 46220 nM T66665 CPM6V1 90645132 IC50 > 100000 nM T66665 CP1OU8 90645133 IC50 = 61230 nM T66665 CBI19Z 90645134 IC50 = 16000 nM T66665 CN4ZE6 90645135 IC50 = 660 nM T66665 C2ZBV6 90645136 IC50 = 1700 nM T66665 C5Z6DG 90645137 IC50 = 1900 nM T66665 CT31LO 90645138 IC50 = 890 nM T66665 CDT1B3 90645139 IC50 = 1300 nM T66665 C62HKB 90645140 IC50 = 470 nM T66665 CU1DO4 90645141 IC50 = 380 nM T66665 CZS0H2 90654426 IC50 = 68200 nM T66665 CEG84Y 90654427 IC50 > 100000 nM T66665 C4B1TH 90654428 IC50 > 100000 nM T66665 CD3AB4 90654429 IC50 > 100000 nM T66665 CC65OW 90654430 IC50 = 46300 nM T66665 C7ZA0W 90654500 IC50 = 110 nM T66665 C2BT3I 90654516 IC50 = 1500 nM T66665 CAMN76 90654517 IC50 = 1200 nM T66665 CSIU57 90654518 IC50 = 26000 nM T66665 CQZT17 90654519 IC50 = 36 nM T66665 C83OSQ 90654520 IC50 = 85 nM T66665 CG4YA1 90654521 IC50 = 53 nM T66665 CT69YE 90656411 IC50 = 18500 nM T66665 CGX4V1 90656412 IC50 = 18200 nM T66665 CL15HG 90656413 IC50 = 20100 nM T66665 CXI32Z 90656414 IC50 = 19200 nM T66665 CR2BL6 90656415 IC50 = 15800 nM T66665 CMLF57 91434450 IC50 = 247 nM T66665 CUFN49 93767862 IC50 > 50000 nM T66665 C4P0DJ 99891916 IC50 = 120 nM T66665 CTF73H 101676817 IC50 = 44500 nM T66665 C6XFT7 101897868 IC50 = 920 nM T66665 CSV2Q7 102532089 IC50 = 20500 nM T66665 C3GKD7 102579754 IC50 = 530 nM T66665 CF5M3K 103954779 IC50 = 10000 nM T66665 C7EOW8 112783730 IC50 = 89 nM T66665 CLI9X6 117072556 IC50 = 50 nM T66665 C0Q1EX 117072557 IC50 = 22800 nM T66665 C9MQW5 118222220 IC50 = 60 nM T66665 C45NGL 118222276 IC50 = 18 nM T66665 C91HFT 118222278 IC50 = 10 nM T66665 C8AMT1 118222288 IC50 = 26 nM T66665 C7YGX4 118222370 IC50 > 10000 nM T66665 C7AYV5 118540795 IC50 = 3650 nM T66665 CC3R1W 118705847 IC50 = 100 nM T66665 CFYD82 118705848 IC50 = 14580 nM T66665 CF7YS2 118705849 IC50 = 8 nM T66665 CTP28O 118705850 IC50 = 15 nM T66665 C46XYG 118705851 IC50 = 59 nM T66665 CP6Q5Z 118705852 IC50 = 51 nM T66665 C25KZC 118705853 IC50 = 110 nM T66665 C8ZP5B 118705854 IC50 = 17810 nM T66665 CH8BD1 118705855 IC50 = 240 nM T66665 C7PU9Q 118706109 IC50 = 140 nM T66665 CZ6P1A 118706110 IC50 = 210 nM T66665 CZ41SY 118706111 IC50 = 41 nM T66665 CAK53T 118706112 IC50 = 67130 nM T66665 CHZQ47 118706113 IC50 = 173600 nM T66665 CO03UN 118706114 IC50 = 1970 nM T66665 CL71XC 118706115 IC50 = 5650 nM T66665 CXZU03 118706116 IC50 = 27090 nM T66665 CI7N0Z 118706117 IC50 = 60980 nM T66665 CA0YD9 118706118 IC50 = 89070 nM T66665 CDPZ58 118706119 IC50 = 95380 nM T66665 CR7PT9 118706120 IC50 = 1320 nM T66665 CFQP30 118706121 IC50 = 530 nM T66665 C49MZI 118706122 IC50 > 500000 nM T66665 CLE92N 118706123 IC50 = 57360 nM T66665 CPR53V 118706201 IC50 = 18550 nM T66665 C9N4TL 118706202 IC50 = 7880 nM T66665 CFW9D7 118706203 IC50 = 9120 nM T66665 CLOT72 118706204 IC50 = 19220 nM T66665 CR46GW 118706205 IC50 = 54320 nM T66665 CWI95H 118706206 IC50 > 100000 nM T66665 CNX45J 118706207 IC50 > 100000 nM T66665 CHP1A7 118706208 IC50 > 100000 nM T66665 CMA91X 118706209 IC50 = 57220 nM T66665 CXY51P 118710092 IC50 > 10000 nM T66665 CC39RL 118710093 IC50 > 10000 nM T66665 C43MCU 118710094 IC50 = 7100 nM T66665 CXE57C 118710095 IC50 = 6800 nM T66665 C7K1CV 118710096 IC50 > 10000 nM T66665 C04UBS 118710097 IC50 > 10000 nM T66665 C0LW4V 118710098 IC50 = 8100 nM T66665 CW9UH2 118710099 IC50 > 10000 nM T66665 CUV78O 118710100 IC50 > 10000 nM T66665 CZHN38 118710101 IC50 > 10000 nM T66665 CY7J3O 118710102 IC50 > 10000 nM T66665 CMP9G8 118710103 IC50 > 10000 nM T66665 C52YJF 118710104 IC50 = 2100 nM T66665 CK2IE6 118710105 IC50 = 3600 nM T66665 CKV43U 118710106 IC50 = 6900 nM T66665 CB5YU6 118710107 IC50 = 10000 nM T66665 CBAQ59 118710108 IC50 = 3400 nM T66665 CSHM97 118710109 IC50 > 10000 nM T66665 C27IGH 118710110 IC50 = 2900 nM T66665 CP2U4A 118710111 IC50 = 10000 nM T66665 C9J8DS 118710112 IC50 = 7200 nM T66665 CSM5I3 118710113 IC50 = 2500 nM T66665 CRA39Z 118710114 IC50 > 10000 nM T66665 CE2J8V 118710115 IC50 = 9500 nM T66665 C50XTM 118710116 IC50 > 10000 nM T66665 C7BAZ1 118710117 IC50 = 6200 nM T66665 CAX96S 118710118 IC50 = 6700 nM T66665 CAZX15 118710119 IC50 = 300 nM T66665 C83UIW 118710120 IC50 = 1800 nM T66665 CZX0H2 118713644 IC50 = 1300 nM T66665 CD35QH 118713753 IC50 = 9900 nM T66665 C1DTY5 118713754 IC50 = 40 nM T66665 CR5WB9 118720945 IC50 = 16 nM T66665 CL2X8K 118721971 IC50 > 5000 nM T66665 CH83RC 118721972 IC50 > 5000 nM T66665 CQ7GX9 118721974 IC50 > 5000 nM T66665 CZ6W4Y 118722547 IC50 = 37660 nM T66665 CFH7X4 118723546 IC50 = 7000 nM T66665 CZDF29 118723547 IC50 = 18000 nM T66665 C1PM6B 118723548 IC50 = 10000 nM T66665 CPJL95 118723549 IC50 = 8000 nM T66665 C6XH0K 118726938 IC50 > 10000 nM T66665 CE7L6H 118726939 IC50 > 10000 nM T66665 CB23OM 118726943 IC50 > 10000 nM T66665 CVU2B8 118726944 IC50 > 10000 nM T66665 C7EU9N 118726945 IC50 > 10000 nM T66665 CMS2J7 118726947 IC50 > 10000 nM T66665 CHM38G 118726948 IC50 > 10000 nM T66665 CY3J0G 118726949 IC50 > 10000 nM T66665 CR6IC4 118726951 IC50 > 10000 nM T66665 C4J5EW 118726952 IC50 > 10000 nM T66665 CVO6Y5 118726954 IC50 > 10000 nM T66665 CA8TS2 118726955 IC50 > 10000 nM T66665 C89LIX 118726956 IC50 > 10000 nM T66665 CIJ62C 118727929 IC50 > 50000 nM T66665 CZ20FX 118727930 IC50 = 8500 nM T66665 C6T7VS 118727931 IC50 > 50000 nM T66665 C0MGP4 118727932 IC50 > 50000 nM T66665 C7CX9E 118727933 IC50 > 50000 nM T66665 CWB87K 118729070 IC50 = 24600 nM T66665 C5YL2D 118729071 IC50 > 100000 nM T66665 CAW2E3 118729078 IC50 > 100000 nM T66665 C12ANV 118729079 IC50 = 68200 nM T66665 C6ZNV4 118729086 IC50 = 17300 nM T66665 CH47SP 118729198 IC50 = 7000 nM T66665 CUH7M2 118729199 IC50 = 4910 nM T66665 C9HS7L 118729200 IC50 = 1070 nM T66665 CYC0M4 118729203 IC50 = 5780 nM T66665 CGAI63 118732322 IC50 = 8340 nM T66665 CSH9W4 118732323 IC50 = 3280 nM T66665 CZ1RW7 118732324 IC50 = 2480 nM T66665 CN0YW1 118732325 IC50 = 2160 nM T66665 CO8EN9 118732326 IC50 = 2630 nM T66665 C1BMZ2 118732327 IC50 = 1120 nM T66665 CGT23L 118732328 IC50 = 11890 nM T66665 C3I0PV 118732329 IC50 = 4830 nM T66665 C32HRJ 118732330 IC50 = 15320 nM T66665 C5FNC2 118732331 IC50 = 4920 nM T66665 C8OS5F 118732332 IC50 = 12680 nM T66665 CI4HR8 118732333 IC50 = 3480 nM T66665 C4I6RK 118732334 IC50 = 26340 nM T66665 CVU70J 118732335 IC50 = 1760 nM T66665 CBEH21 118732336 IC50 = 18260 nM T66665 CH7Y4R 118732337 IC50 = 32260 nM T66665 CF1Z6J 118732338 IC50 = 3660 nM T66665 CG01BT 118732339 IC50 = 460 nM T66665 CH4XL0 118732340 IC50 = 330 nM T66665 C3WTD0 118732341 IC50 = 1020 nM T66665 C6YXJ5 118732342 IC50 = 7240 nM T66665 C87MQF 118732343 IC50 = 2280 nM T66665 CCEO82 118732344 IC50 = 8240 nM T66665 CW79HI 118732345 IC50 = 1260 nM T66665 C48ZGB 118732346 IC50 = 6880 nM T66665 CC57TX 118732347 IC50 = 2740 nM T66665 CNY30X 118732348 IC50 = 16270 nM T66665 CH8R9Z 118736803 IC50 = 2520 nM T66665 CKI03L 118736804 IC50 = 6040 nM T66665 C2R8CP 118736805 IC50 = 8240 nM T66665 CL0SV1 118736806 IC50 = 6020 nM T66665 C9C2TL 118736807 IC50 = 13700 nM T66665 C9GB1Z 118736808 IC50 = 8600 nM T66665 C4EB9O 118736809 IC50 = 17800 nM T66665 CCBQ34 118736810 IC50 = 9700 nM T66665 CG1AW4 118736811 IC50 = 1300 nM T66665 CEU29Z 118736812 IC50 = 2500 nM T66665 C3A9EQ 118736813 IC50 = 2700 nM T66665 C0K2AH 118855478 IC50 = 970 nM T66665 CILM06 121423933 IC50 > 10000 nM T66665 CN5CA4 121427628 IC50 > 10000 nM T66665 CVRP92 122177370 IC50 = 890 nM T66665 CXP9U8 122177371 Ki = 5 nM T66665 CJ9D1Q 122177372 IC50 = 21310 nM T66665 C0CMT2 122177373 Ki = 12 nM T66665 CR35MW 122177374 Ki = 4659 nM T66665 C27WEH 122177375 IC50 = 1000 nM T66665 C7WZ0I 122177376 IC50 = 6.3 nM T66665 C45ZRD 122177377 IC50 = 2500 nM T66665 C0CIM4 122177378 Ki = 1342 nM T66665 CDX51K 122177379 IC50 = 8330 nM T66665 CCO72V 122177380 Ki = 983 nM T66665 CG08QN 122177381 IC50 = 970 nM T66665 CD7BH4 122177382 IC50 = 10310 nM T66665 CNJ7Y1 122177383 IC50 = 47 nM T66665 C0T8UG 122177384 IC50 = 6610 nM T66665 CQCH60 122177385 IC50 = 13500 nM T66665 C3CKO7 122178781 IC50 = 6400 nM T66665 CK3O4I 122182704 IC50 = 1700 nM T66665 CK6AX3 122182705 IC50 = 2600 nM T66665 CKF4H7 122182706 IC50 = 1800 nM T66665 CJ8D7T 122182707 IC50 = 10500 nM T66665 CJ6E4Z 122182708 IC50 = 4700 nM T66665 C5I8SH 122182709 IC50 = 4100 nM T66665 C1VE5G 122182710 IC50 = 6800 nM T66665 C9CE7G 122182711 IC50 = 9900 nM T66665 CW14SV 122182712 IC50 = 5900 nM T66665 CGX21Y 122182713 IC50 = 3900 nM T66665 CL6K3X 122184817 IC50 = 890 nM T66665 C7NR8C 122184818 IC50 = 220 nM T66665 C61DMQ 122184819 IC50 = 280 nM T66665 CI4OQ5 122192740 IC50 = 12000 nM T66665 CP90JH 122192741 IC50 > 100000 nM T66665 CU96HS 122192742 IC50 > 100000 nM T66665 C5Z4RW 122192743 IC50 > 100000 nM T66665 CKZD31 122393225 IC50 = 20 nM T66665 C1B9FQ 122603295 IC50 = 279 nM T66665 CDN0A3 123278303 IC50 > 10000 nM T66665 C70SYK 126842939 IC50 = 860 nM T66665 CVJ01U 127029897 IC50 > 100000 nM T66665 C8M0JF 127029898 IC50 = 730 nM T66665 CJO07B 127030237 IC50 = 1400 nM T66665 CAIQ36 127030238 IC50 = 200 nM T66665 C6UZ2W 127030243 IC50 = 850 nM T66665 CYM16I 127031160 IC50 > 100000 nM T66665 CTVI73 127031161 IC50 = 560 nM T66665 CN4I7Q 127031735 IC50 = 13000 nM T66665 C5D7HI 127033540 IC50 > 100000 nM T66665 C1BNI4 127033589 IC50 = 690 nM T66665 CGJ2W4 127033590 IC50 = 930 nM T66665 CUB06J 127033591 IC50 = 12100 nM T66665 CWF6D9 127034425 IC50 = 13000 nM T66665 CK3F1Z 127034778 IC50 = 1750 nM T66665 C4HR7O 127035271 IC50 = 3980 nM T66665 CK5U1E 127035272 IC50 = 4710 nM T66665 CN5WP7 127035406 IC50 = 2170 nM T66665 C7O5FJ 127035407 IC50 = 3740 nM T66665 C0PJ1F 127035408 IC50 = 5940 nM T66665 CFMX84 127035409 IC50 = 1160 nM T66665 CT2S1D 127035755 IC50 = 980 nM T66665 CX17OE 127035756 IC50 = 2840 nM T66665 CNO5S9 127035770 IC50 = 1620 nM T66665 C5T8PA 127035771 IC50 = 3410 nM T66665 CAXB08 127035772 IC50 = 2670 nM T66665 C9A4YS 127035963 IC50 = 1760 nM T66665 CM76EF 127035964 IC50 = 2110 nM T66665 C1NL5H 127035965 IC50 = 1980 nM T66665 C0TX4B 127036337 IC50 = 4670 nM T66665 C94INO 127037903 IC50 = 1520 nM T66665 C5KUY4 127037904 IC50 = 2640 nM T66665 C38DAI 127037905 IC50 = 560 nM T66665 C47MSQ 127037906 IC50 = 1970 nM T66665 C2T5LW 127038271 IC50 = 6340 nM T66665 C12SUP 127038624 IC50 > 1000 nM T66665 C7QLE4 127040263 IC50 = 970 nM T66665 C8NJD4 127041577 IC50 = 3560 nM T66665 C2JQI4 127041578 IC50 = 2110 nM T66665 CYMJ97 127041579 IC50 = 1840 nM T66665 CNOW51 127041580 IC50 = 1430 nM T66665 CBF6E9 127041850 IC50 > 1000 nM T66665 C1F8IA 127042131 IC50 = 10300 nM T66665 C1WF9X 127042132 IC50 = 1000 nM T66665 CZI8L4 127042820 IC50 = 4130 nM T66665 CVMZ36 127042821 IC50 = 6110 nM T66665 CW1Y3E 127042822 IC50 = 3650 nM T66665 CYNS97 127042823 IC50 = 6110 nM T66665 CT1V2C 127042824 IC50 = 3890 nM T66665 C1PF5U 127042828 IC50 = 1980 nM T66665 C9XK8Q 127043035 IC50 = 80 nM T66665 CU0Z5F 127043036 IC50 = 50 nM T66665 C2RJU9 127043217 IC50 = 300 nM T66665 C29WPZ 127043218 IC50 = 56000 nM T66665 C4ZI6F 127043222 IC50 = 20000 nM T66665 C4LD1B 127044382 IC50 = 8000 nM T66665 CYF3S4 127045511 IC50 = 22000 nM T66665 CO4YJ7 127045512 IC50 = 8000 nM T66665 CK3SV9 127045513 IC50 = 19000 nM T66665 CQA34G 127049134 IC50 = 4530 nM T66665 CV64AJ 127049135 IC50 = 6940 nM T66665 CRO71E 127049136 IC50 = 4790 nM T66665 CXMV19 127049150 IC50 = 10410 nM T66665 C8F3NJ 127049474 IC50 = 21930 nM T66665 C3VK2H 127051106 IC50 = 8830 nM T66665 CZ3M1S 127051109 IC50 = 1060 nM T66665 CTW94N 127051121 IC50 = 540 nM T66665 CT96YA 127051122 IC50 = 300 nM T66665 C9U5CW 127051123 IC50 = 470 nM T66665 CAQD52 127051124 IC50 = 260 nM T66665 CJQM74 127051125 IC50 = 170 nM T66665 C1NB2H 127051922 IC50 = 7130 nM T66665 C6OBL0 127051923 IC50 = 6250 nM T66665 CB96YL 127051924 IC50 = 10360 nM T66665 C64RNC 127051925 IC50 = 6090 nM T66665 CNH54C 127052535 IC50 = 130 nM T66665 C62ZJO 127052536 IC50 = 90 nM T66665 CO4QG9 129886428 IC50 = 90 nM T66665 C5T4EQ 131801158 IC50 = 230 nM T66665 CL9SH5 132495362 IC50 = 9230 nM T66665 C4L6UZ 132547258 IC50 = 4440 nM T66665 CGBR54 132547259 IC50 = 300 nM T66665 CW4MP2 132547260 IC50 = 330 nM T66665 CUFI36 132603679 IC50 = 35500 nM T66665 CQ6ZR1 132603681 IC50 = 4700 nM T66665 C9XT2A 132607269 Ki = 920 nM T66665 CQO23I 134131456 IC50 = 4580 nM T66665 CGR8K3 134132260 IC50 = 15120 nM T66665 C51BVC 134132774 IC50 = 20000 nM T66665 C43OPG 134134531 IC50 = 8280 nM T66665 C19USV 134134738 IC50 = 281838.29 nM T66665 CQK60R 134135733 IC50 = 269153.48 nM T66665 C82SJP 134136283 IC50 = 10710 nM T66665 CFM0C9 134138215 IC50 = 9120 nM T66665 CAEZ47 134138298 IC50 = 218776.16 nM T66665 CD07XW 134139182 IC50 > 1000 nM T66665 CY75JU 134139783 IC50 = 14120 nM T66665 CI97WR 134140189 IC50 > 1000 nM T66665 C90LTZ 134141655 IC50 = 245470.89 nM T66665 CV8D2I 134141804 IC50 = 6890 nM T66665 C6U7LZ 134143054 IC50 = 303400 nM T66665 CGHI39 134143639 IC50 = 10230 nM T66665 CR5I2D 134144193 IC50 = 8320 nM T66665 C92HTQ 134144693 IC50 = 16120 nM T66665 CH86VI 134147676 IC50 = 459000 nM T66665 CJTO28 134149141 IC50 = 7950 nM T66665 C5XR2B 134152086 IC50 = 4570881.9 nM T66665 CJI9Y3 134152691 IC50 = 251188.64 nM T66665 CDV05U 134154144 IC50 = 295120.92 nM T66665 CA08HM 134154737 IC50 = 129900 nM T66665 CTQ0D6 134155386 IC50 = 12570 nM T66665 C7UHV2 134156637 IC50 = 11020 nM T66665 C1GY2T 135156251 EC50 > 10000 nM T66665 CHS9Q1 135401075 IC50 = 27000 nM T66665 CZ0M4A 135407197 IC50 > 20000 nM T66665 C5AXQ9 135411265 IC50 = 1100 nM T66665 C5XLH3 135412819 IC50 = 47000 nM T66665 C6Z1ME 135417317 IC50 > 20000 nM T66665 CB2L3G 135419219 IC50 = 64 nM T66665 CPTI38 135419252 IC50 = 6500 nM T66665 CTIX57 135428092 IC50 = 32410 nM T66665 CN3KQ5 135430565 IC50 = 55000 nM T66665 CVR89H 135444615 IC50 = 140 nM T66665 C1PMI3 135444631 IC50 = 1700 nM T66665 CMQ2F9 135458830 IC50 = 1020 nM T66665 C10NPU 135461834 IC50 > 20000 nM T66665 C6P7QT 135464202 IC50 = 1500 nM T66665 CPEX68 135467810 IC50 > 20000 nM T66665 C28NZL 135467819 IC50 > 20000 nM T66665 C6HYD1 135474341 IC50 = 100000 nM T66665 CJD1E8 135476136 IC50 > 20000 nM T66665 CA8UC6 135476177 IC50 > 20000 nM T66665 C4HW1Z 135480072 IC50 = 570 nM T66665 CQ29PT 135480085 IC50 = 2700 nM T66665 C8JH3G 135491761 IC50 = 9400 nM T66665 CH9C7U 135493485 IC50 > 20000 nM T66665 C8XMC3 135493549 IC50 > 20000 nM T66665 CSB0M9 135494223 IC50 = 9700 nM T66665 CE76OB 135497218 IC50 = 6100 nM T66665 CZOP78 135497261 IC50 = 41000 nM T66665 C9CT1H 135502784 IC50 < 20000 nM T66665 CU53ZB 135503592 IC50 > 20000 nM T66665 CK6C8G 135503854 IC50 = 100000 nM T66665 CAB5M3 135503855 IC50 > 20000 nM T66665 CWN8H2 135506078 IC50 = 79000 nM T66665 C5RYH6 135512019 IC50 = 3200 nM T66665 C9TZ2E 135513737 IC50 > 20000 nM T66665 C5Z9ED 135513895 IC50 = 3000 nM T66665 CW7YI3 135513937 IC50 > 20000 nM T66665 CL28MS 135515182 IC50 = 19000 nM T66665 CZ4T5K 135518175 IC50 = 3500 nM T66665 C3V1HA 135524515 IC50 > 20000 nM T66665 CDC4X5 135525549 IC50 = 11500 nM T66665 C6VO2S 135529786 IC50 > 20000 nM T66665 C2DUW6 135529925 IC50 > 20000 nM T66665 CX9H1L 135532444 IC50 > 100000 nM T66665 CCG7O5 135537152 IC50 = 26000 nM T66665 C2VFX1 135543599 IC50 = 15450 nM T66665 CH6TK3 135543992 IC50 = 1400 nM T66665 C12FNX 135637726 IC50 = 6490 nM T66665 CU0OW5 135693491 IC50 = 7.2 nM T66665 C2YX9D 135748955 IC50 = 47 nM T66665 CF1W0U 135783304 IC50 = 262000 nM T66665 C8K2NT 135786528 IC50 = 11000 nM T66665 CT1C9J 135786531 IC50 = 4100 nM T66665 C3ACW8 135786533 IC50 > 20000 nM T66665 CGBM73 135786534 IC50 > 20000 nM T66665 C1S6KC 135786539 IC50 = 23000 nM T66665 C7OJC8 135786549 IC50 = 1300 nM T66665 C8JCM5 135786553 IC50 = 17000 nM T66665 CX25SL 135786554 IC50 = 9600 nM T66665 C5KLO4 135905678 IC50 = 18960 nM T66665 C3N2FJ 135906278 IC50 > 10000 nM T66665 C1XQY2 135923992 IC50 = 10710 nM T66665 CHM3Y8 135972420 IC50 = 2000 nM T66665 CZMT92 136029176 IC50 = 240 nM T66665 CJ5S1X 136029177 IC50 = 550 nM T66665 CK09XP 136036210 IC50 > 50000 nM T66665 CXG07W 136042393 IC50 = 11600 nM T66665 C2R9VH 136044097 IC50 = 410 nM T66665 CYSW23 136094858 IC50 = 7570 nM T66665 CFO48N 136094859 IC50 = 9970 nM T66665 CM8Q9X 136152995 IC50 = 2710 nM T66665 C5T2VU 136152996 IC50 = 20284298.83 nM T66665 C51PHR 136152997 IC50 = 12594473.01 nM T66665 CNM2Z3 136211082 IC50 = 14000 nM T66665 CW4J5O 136224196 IC50 = 5130 nM T66665 C94ZVL 136240270 IC50 = 7110 nM T66665 C1WOF5 136241419 IC50 = 8800 nM T66665 C4KTV2 136241451 IC50 = 360 nM T66665 C8Z7XM 136241655 IC50 = 400 nM T66665 CJ1FC5 136245110 IC50 = 7500 nM T66665 CC8Q4G 136264297 IC50 = 7000 nM T66665 C56NTX 136264298 IC50 = 520 nM T66665 CSK95Y 136504263 IC50 = 13 nM T66665 CRT4Q2 136961752 IC50 = 970 nM T66665 C2IPJ1 137412816 IC50 = 190 nM T66665 CCYO27 137412823 IC50 = 8 nM T66665 C52PCB 137412826 IC50 = 46 nM T66665 C9G2IS 137412832 IC50 > 10000 nM T66665 C9K7QT 137412863 IC50 > 100000 nM T66665 C34NHP 137631356 IC50 = 1720 nM T66665 CNE1Y9 137631969 IC50 = 6 nM T66665 C4LD8H 137632223 IC50 = 16.2 nM T66665 CBEZ81 137632289 IC50 = 1830 nM T66665 CX29BF 137632390 IC50 = 450 nM T66665 C02ZKT 137632796 IC50 = 2500 nM T66665 C2FA0K 137632978 IC50 = 540 nM T66665 C2ROQ9 137633369 IC50 = 2780 nM T66665 C1GN8O 137633399 IC50 = 2810 nM T66665 C7OP3D 137634032 IC50 = 1400 nM T66665 C0LYA4 137634609 IC50 = 1430 nM T66665 CMH92C 137635036 IC50 = 302 nM T66665 CED48F 137635504 IC50 = 550 nM T66665 CL02CU 137636006 IC50 = 870 nM T66665 C0QPM3 137636484 IC50 = 4500 nM T66665 C0ZTQ4 137637033 IC50 = 2540 nM T66665 CGP8S7 137637113 IC50 = 740 nM T66665 CC53HT 137637798 IC50 = 290 nM T66665 CXU5M3 137638275 IC50 = 1750 nM T66665 C72SBZ 137638298 IC50 > 10000 nM T66665 CJ76FA 137638345 IC50 = 300 nM T66665 CMNL79 137638584 IC50 = 1860 nM T66665 C4WX2T 137638629 IC50 = 6930 nM T66665 CS8KB1 137638984 IC50 = 20.1 nM T66665 CG16DR 137638994 IC50 > 10000 nM T66665 C6T1GM 137639040 IC50 = 910 nM T66665 CF12ZY 137639045 IC50 = 1210 nM T66665 C8DGE3 137639285 IC50 = 56 nM T66665 C9ZXE6 137639615 IC50 = 360 nM T66665 CP1I9Z 137639679 IC50 = 490 nM T66665 CR8YQ0 137639813 IC50 = 190 nM T66665 C2GEU5 137639906 IC50 > 10000 nM T66665 CP59LO 137640049 IC50 = 1170 nM T66665 CCY7B8 137640363 IC50 > 10000 nM T66665 CGQD73 137640436 IC50 = 520 nM T66665 C0PL9E 137640952 IC50 = 110 nM T66665 CGQ04J 137641089 IC50 = 90.1 nM T66665 C95HDN 137641244 IC50 = 680 nM T66665 CYV07I 137642019 IC50 = 181 nM T66665 CEYG80 137642209 IC50 > 10000 nM T66665 CAJ5V9 137642414 IC50 = 1450 nM T66665 CG23XO 137642954 IC50 = 1410 nM T66665 C7MLV2 137643935 IC50 = 1610 nM T66665 CBP1L2 137644202 IC50 = 690 nM T66665 C91WXG 137644775 IC50 = 1910 nM T66665 CPVY52 137644807 IC50 = 670 nM T66665 C5QG8C 137645786 IC50 = 4200 nM T66665 CQK8H9 137646026 IC50 = 230 nM T66665 CY70NF 137646137 IC50 = 1120 nM T66665 CZVW72 137647065 IC50 = 1120 nM T66665 CZT65P 137647326 IC50 = 490 nM T66665 C1R9QE 137647998 IC50 = 2330 nM T66665 C14TRW 137648756 IC50 = 1670 nM T66665 CZ0U9Q 137648775 IC50 = 1980 nM T66665 C1SOP6 137649486 IC50 = 400 nM T66665 CC7X5E 137649564 IC50 = 6600 nM T66665 C6NES9 137649621 IC50 = 1760 nM T66665 CK86ZB 137649633 IC50 = 110 nM T66665 CJHR31 137649745 IC50 = 3360 nM T66665 CHJ07Q 137649937 IC50 = 340 nM T66665 COZ38A 137650099 IC50 = 780 nM T66665 CSO31J 137650735 IC50 = 1280 nM T66665 C4PUJ6 137650894 IC50 = 1960 nM T66665 C29KWG 137650898 IC50 = 770 nM T66665 CDFH04 137652081 IC50 = 3540 nM T66665 C3LJY7 137652097 IC50 = 100 nM T66665 CILT87 137652137 IC50 = 430 nM T66665 C3CA7S 137652330 IC50 = 440 nM T66665 CXFT57 137652461 IC50 = 1130 nM T66665 C87VSD 137652535 IC50 = 820 nM T66665 C81HNM 137652647 IC50 = 1910 nM T66665 CN63WS 137652773 IC50 = 560 nM T66665 C7WR8J 137653640 IC50 = 1630 nM T66665 C2MP0H 137653651 IC50 = 160 nM T66665 C2D6KC 137653913 IC50 = 780 nM T66665 CE4RY1 137654190 IC50 = 330 nM T66665 CCK5E0 137655831 IC50 = 1550 nM T66665 CW58SX 137656317 IC50 = 780 nM T66665 C5N1TZ 137657786 IC50 = 3140 nM T66665 C4EG5U 137658493 IC50 = 1690 nM T66665 CT29JI 137658900 IC50 = 6880 nM T66665 C1ONT8 137659426 IC50 = 860 nM T66665 C24EJC 137659682 IC50 = 2860 nM T66665 C7NE9X 137659718 IC50 > 10000 nM T66665 CIYT80 137659915 IC50 = 170 nM T66665 C2HT5O 137659979 IC50 = 310 nM T66665 C23FQJ 137660504 IC50 = 1220 nM T66665 CY0FH9 137660585 IC50 = 1740 nM T66665 C45IKL 137660851 IC50 = 330 nM T66665 CPAL37 137661149 IC50 = 3290 nM T66665 C1MKL9 137661257 IC50 = 490 nM T66665 C80LGK 137661666 IC50 = 9580 nM T66665 C20HZY 137661944 IC50 = 1490 nM T66665 CF74TS 137661963 IC50 = 530 nM T66665 CQS3W7 137662098 IC50 = 2110 nM T66665 CM3UF7 137700779 IC50 > 10000 nM T66665 C2OQN1 138115373 IC50 > 100000 nM T66665 CX06CI 138542656 IC50 > 50000 nM T66665 CX0L1A 139035063 IC50 = 420 nM T66665 C7N9PX 139188449 IC50 = 1870 nM T66665 CQZ84L 139188450 IC50 = 930 nM T66665 C3Y9MC 144673436 IC50 = 180 nM T66665 CIT37B 145949529 IC50 = 60000 nM T66665 C3ZFV8 145949611 IC50 = 270 nM T66665 CHA86D 145949872 IC50 = 7000 nM T66665 C51VOJ 145949898 IC50 = 500 nM T66665 C5XGJ0 145949944 IC50 = 45300 nM T66665 CFNO28 145950339 IC50 = 790 nM T66665 CW5NG1 145950458 IC50 = 500 nM T66665 CG37FR 145950583 IC50 = 280 nM T66665 CI02OR 145950689 IC50 = 600 nM T66665 CK8TQ0 145951126 IC50 = 600 nM T66665 C2B6JH 145951867 IC50 = 70000 nM T66665 C19FCR 145952084 IC50 = 7150 nM T66665 CL6X8E 145952627 IC50 = 14500 nM T66665 CCN16Y 145952805 IC50 = 910 nM T66665 CE4R1P 145952838 IC50 = 5320 nM T66665 CMI93X 145952895 IC50 = 12490 nM T66665 C2FVO7 145953074 IC50 = 810 nM T66665 CWQ40O 145954141 IC50 = 80 nM T66665 C7HK6U 145954201 IC50 = 2150 nM T66665 C46FPD 145954463 IC50 = 56400 nM T66665 CJ67ER 145954492 IC50 = 80 nM T66665 CMW75D 145954530 IC50 = 34600 nM T66665 C4TXP8 145954758 IC50 = 480 nM T66665 CP0KQ3 145954913 IC50 = 40 nM T66665 C0C9PE 145955075 IC50 = 75000 nM T66665 C3A1GS 145955474 IC50 = 60 nM T66665 CS5B3U 145955705 IC50 = 70000 nM T66665 CI4YB1 145956104 IC50 = 100 nM T66665 CR05AN 145956878 IC50 = 12800 nM T66665 CS40VG 145957891 IC50 = 100000 nM T66665 C19TPY 145958203 IC50 = 970 nM T66665 CIS8Y7 145958302 IC50 = 500 nM T66665 C3FW1B 145958377 IC50 = 6000 nM T66665 CI4PU9 145958703 IC50 = 1000 nM T66665 CZ2X3O 145959205 IC50 = 6000 nM T66665 CMR4P6 145959224 IC50 = 3140 nM T66665 CBL1V0 145959229 IC50 = 3100 nM T66665 C1BLR8 145959460 IC50 = 580 nM T66665 C35AQV 145960574 IC50 = 80000 nM T66665 C7F1WN 145960726 IC50 = 390 nM T66665 C6R3AF 145960841 IC50 = 310 nM T66665 CZE9D3 145960993 IC50 = 6000 nM T66665 CRV1U7 145962585 IC50 = 310 nM T66665 CBG7X0 145963101 IC50 = 310 nM T66665 C65QKS 145963415 IC50 = 310 nM T66665 CYX01T 145966366 IC50 = 45540 nM T66665 CPR90E 145969152 IC50 = 7461 nM T66665 CUXQ13 145971245 IC50 = 880 nM T66665 C8U9TX 145971276 IC50 = 340 nM T66665 CO4T7E 145971990 IC50 = 90000 nM T66665 C8V1TL 145972167 IC50 = 100000 nM T66665 C2EYD6 145972696 IC50 = 6420 nM T66665 CUG3W4 145978901 IC50 = 9500 nM T66665 CR96QC 145978940 IC50 > 100000 nM T66665 C9EVJ0 145979118 IC50 = 540 nM T66665 CFZ9E6 145979142 IC50 = 13777 nM T66665 C7ZOM8 145979619 IC50 = 12610 nM T66665 CKO46M 145979761 IC50 > 100000 nM T66665 CE8Z4M 145979875 IC50 = 110 nM T66665 C9H6AW 145979979 IC50 = 18320 nM T66665 CS85AP 145980216 IC50 = 21780 nM T66665 C6DYF0 145980296 IC50 > 100000 nM T66665 CV24IQ 145980499 IC50 = 370 nM T66665 CS2E7V 145981172 IC50 > 100000 nM T66665 CO72CD 145981197 IC50 = 170 nM T66665 CIZ20X 145981840 IC50 = 840 nM T66665 C9MSG2 145982141 IC50 > 100000 nM T66665 CXO6V1 145982200 IC50 = 890 nM T66665 CASB43 145982402 IC50 = 81200 nM T66665 CZPC04 145982667 IC50 = 1190 nM T66665 CJGE56 145982912 IC50 = 670 nM T66665 C0LU3T 145982976 IC50 = 1080 nM T66665 C20AWS 145983008 IC50 = 5020 nM T66665 CA8U6O 145983125 IC50 = 2120 nM T66665 CGZ73L 145983279 IC50 = 1410 nM T66665 CR61XP 145983281 IC50 = 4800 nM T66665 CP54SE 145983381 IC50 = 230 nM T66665 C0HE8J 145983476 IC50 = 1210 nM T66665 C2W1PX 145983528 IC50 = 1390 nM T66665 CMTE25 145983596 IC50 = 4790 nM T66665 C0LF5R 145983962 IC50 = 1660 nM T66665 CAB1M0 145984018 IC50 = 350 nM T66665 CDW7Q2 145984214 IC50 = 6830 nM T66665 C09ZYR 145984318 IC50 = 2200 nM T66665 C6TD4Z 145984372 IC50 = 770 nM T66665 C6RS2D 145984423 IC50 = 3530 nM T66665 CUY3T9 145984477 IC50 = 4330 nM T66665 CB9X6S 145984519 IC50 = 5940 nM T66665 C8-MAR-07 145984539 IC50 = 4430 nM T66665 CA3PM5 145984912 IC50 = 38160 nM T66665 CXPK46 145984992 IC50 = 2120 nM T66665 C3KEW1 145985004 IC50 = 1360 nM T66665 C50TGP 145985054 IC50 = 2540 nM T66665 C1LEX8 145985067 IC50 = 1440 nM T66665 CTE68V 145985355 IC50 = 8580 nM T66665 CRIT31 145985451 IC50 = 540 nM T66665 CL6ZW3 145985573 IC50 = 422 nM T66665 CG0S8Q 145985628 IC50 = 670 nM T66665 C7FWH1 145985695 IC50 = 930 nM T66665 C1T2XR 145985744 IC50 = 420 nM T66665 C2RO7H 145986163 IC50 = 2840 nM T66665 CBEG25 145986220 IC50 = 1770 nM T66665 CV6BD5 145986241 IC50 = 5020 nM T66665 C9MI3W 145986376 IC50 = 180 nM T66665 CHD9A0 145986886 IC50 = 240 nM T66665 C45FWQ 145987526 IC50 = 160 nM T66665 CKOF74 145987835 IC50 = 340 nM T66665 CGO94I 145987940 IC50 = 4170 nM T66665 CFV56O 145988248 IC50 = 10790 nM T66665 CUC8A2 145988507 IC50 = 630 nM T66665 CEL6S3 145988681 IC50 = 250 nM T66665 C9D1VG 145988772 IC50 = 1340 nM T66665 CN6WV5 145989076 IC50 = 1020 nM T66665 C35VEG 145989087 IC50 = 19730 nM T66665 C6DN9E 145989219 IC50 = 16210 nM T66665 CNS6C2 145989313 IC50 > 100000 nM T66665 CEQ37S 145989981 IC50 = 42 nM T66665 CVU8N9 145990110 IC50 = 57 nM T66665 CEQ79N 145990431 IC50 = 1340 nM T66665 CC3YU0 145990700 IC50 = 250 nM T66665 CT63IW 145991059 IC50 = 1330 nM T66665 CPO62F 145991413 IC50 = 560 nM T66665 CM7BD5 145991610 IC50 = 520 nM T66665 C17YJO 145991798 IC50 = 890 nM T66665 CW3UG5 145992883 IC50 = 8145 nM T66665 CZ0J6H 145992911 IC50 = 11050 nM T66665 C4QK6J 145992976 IC50 = 560 nM T66665 C1TM3J 145993175 IC50 = 650 nM T66665 CW91DU 145993284 IC50 = 960 nM T66665 C87MDX 145994033 IC50 = 351 nM T66665 CY43GM 145994107 IC50 = 1040 nM T66665 CTI1A7 149810461 IC50 = 870 nM T66665 CM32VY 150503533 IC50 = 310 nM T66665 C43PXH 151104161 IC50 = 640 nM T66665 CC6XK3 151319427 IC50 = 160 nM T66665 C89BKF 153320917 IC50 > 50000 nM T66665 CB68HZ 153320918 IC50 = 300 nM T66665 CJ2LT9 155490749 IC50 = 23.3 nM T66665 CK07AV 155490796 IC50 = 21.86 nM T66665 CFP09E 155510363 IC50 = 1050 nM T66665 CGR20J 155510471 IC50 = 260 nM T66665 CU5E9G 155511187 IC50 = 18.35 nM T66665 CS86EI 155511524 IC50 = 150 nM T66665 CCIZ41 155512205 IC50 = 108.3 nM T66665 C3JX1B 155512689 IC50 = 250 nM T66665 C3R8LP 155512734 IC50 = 56.17 nM T66665 CA7M4W 155513070 IC50 = 420 nM T66665 CYXQ71 155513215 IC50 = 110 nM T66665 C3UQ9M 155513357 IC50 = 23.21 nM T66665 CP6N7G 155513887 IC50 = 210 nM T66665 C8BYT1 155514150 IC50 = 380 nM T66665 C5AF0O 155514534 IC50 = 970 nM T66665 CM0OK6 155514659 IC50 = 1250 nM T66665 CZB64G 155514739 IC50 = 830 nM T66665 CAZ16P 155514890 IC50 = 210 nM T66665 CJO5Y4 155514909 IC50 = 110 nM T66665 C7U8HX 155515015 IC50 = 1110 nM T66665 CK21YX 155515749 IC50 = 15.56 nM T66665 CH41WR 155516265 IC50 = 430000 nM T66665 CM0O8D 155516306 IC50 = 1000 nM T66665 CFD4A0 155516566 IC50 = 600 nM T66665 C5VNH3 155516647 IC50 = 1880 nM T66665 CY3DR9 155516693 IC50 = 39.43 nM T66665 CK2R8I 155516851 IC50 = 10100 nM T66665 CNR04X 155517006 IC50 = 110 nM T66665 CJKZ29 155517041 IC50 = 210 nM T66665 CHT40W 155517183 IC50 = 60 nM T66665 C3P4MO 155517441 IC50 = 48.79 nM T66665 CXGS50 155517610 IC50 = 650000 nM T66665 CQK2J3 155518007 IC50 = 170 nM T66665 CP9W0Z 155518171 IC50 = 360 nM T66665 C02FZA 155519294 IC50 = 230 nM T66665 CCH5E8 155519683 IC50 = 2790 nM T66665 CD8NP7 155519869 IC50 = 7590 nM T66665 C64JSW 155520540 IC50 = 330 nM T66665 CL4ZA7 155520575 IC50 > 50000 nM T66665 C5I3OE 155520725 IC50 = 130 nM T66665 C02HAV 155521349 IC50 = 1930 nM T66665 C5BH7V 155521378 IC50 = 520 nM T66665 CA0R9H 155521417 IC50 = 540000 nM T66665 CVI9A4 155521418 IC50 = 290 nM T66665 CQ3N6D 155521710 IC50 = 82.99 nM T66665 CPKS90 155521809 IC50 = 2800 nM T66665 C98MBO 155522237 IC50 = 2110 nM T66665 C69GCU 155522308 IC50 = 7530 nM T66665 CB41LZ 155522446 IC50 = 210 nM T66665 CSY34V 155523202 IC50 = 122.8 nM T66665 C97MPO 155523342 IC50 = 460000 nM T66665 C4PGA5 155523362 IC50 = 1490 nM T66665 CA8Q1L 155523402 IC50 = 1100 nM T66665 C70URH 155523591 IC50 = 410 nM T66665 CF82YG 155523642 IC50 = 1650 nM T66665 C15FBJ 155524017 IC50 = 330 nM T66665 C69ECX 155524453 IC50 = 44100 nM T66665 CQ4MB8 155524522 IC50 = 910 nM T66665 CM37UN 155524616 IC50 = 120 nM T66665 CO1KL9 155524670 IC50 = 10100 nM T66665 CSB47U 155524970 IC50 = 100 nM T66665 CX36AH 155526366 IC50 = 690 nM T66665 CYI18A 155526372 IC50 = 400 nM T66665 CC1LR8 155526446 IC50 = 1950 nM T66665 C30OZI 155527652 IC50 = 13310 nM T66665 CK7EU9 155527685 IC50 = 43000 nM T66665 C8U4BP 155527852 IC50 = 5470 nM T66665 CE0J1Y 155528353 IC50 > 500000 nM T66665 CME0N2 155528406 IC50 = 120 nM T66665 CS3Z9A 155528460 IC50 > 200000 nM T66665 C80BRK 155528880 IC50 = 190 nM T66665 CB9M1X 155529539 IC50 = 4690 nM T66665 C2GLH7 155529640 IC50 = 5200 nM T66665 C7ZA5P 155530097 IC50 = 250 nM T66665 CB4WF1 155530728 IC50 = 19.77 nM T66665 C8JZH5 155530824 IC50 = 1280 nM T66665 C1QXU2 155530946 IC50 = 61.24 nM T66665 CTS30K 155530971 IC50 = 2990 nM T66665 C1VYC9 155531564 IC50 = 50 nM T66665 CIJ3G0 155531569 IC50 = 920 nM T66665 C51EJF 155531595 IC50 = 1250 nM T66665 CUL96H 155531758 IC50 = 89.8 nM T66665 CX7Y0S 155531849 IC50 > 50000 nM T66665 CRD14L 155532032 IC50 = 189.77 nM T66665 C2HMZ3 155532215 IC50 = 10100 nM T66665 CCQE28 155532511 IC50 = 310 nM T66665 CD4YR2 155533161 IC50 > 300000 nM T66665 C9J0RH 155534497 IC50 > 50000 nM T66665 CD94TA 155534770 IC50 = 14 nM T66665 C6RB5J 155534811 IC50 = 10790 nM T66665 C7QL5Y 155534969 IC50 = 38000 nM T66665 CA69IG 155534995 IC50 = 4240 nM T66665 C8CG4Z 155535032 IC50 = 10000 nM T66665 CE3VB4 155535321 IC50 = 45400 nM T66665 CWK2R1 155535482 IC50 = 140 nM T66665 CA3GN2 155535611 IC50 = 2250 nM T66665 CBQI97 155536239 IC50 = 2000 nM T66665 CO2TU1 155536282 IC50 = 560 nM T66665 CDC36T 155536309 IC50 = 600 nM T66665 C2PN5F 155536316 IC50 = 44000 nM T66665 CA15BW 155536520 IC50 = 20 nM T66665 CGV02Q 155536953 IC50 = 100 nM T66665 CJ97NX 155536975 IC50 = 100 nM T66665 CLS7Q9 155537343 IC50 = 450000 nM T66665 C2Z7GX 155537370 IC50 = 43800 nM T66665 CN4PC5 155537482 IC50 = 100 nM T66665 CD4F8L 155537530 IC50 = 10100 nM T66665 CA05NV 155537808 IC50 = 3570 nM T66665 CY91IQ 155538558 IC50 = 190 nM T66665 CN5G0R 155538929 IC50 > 50000 nM T66665 C9H0JX 155539820 IC50 = 890 nM T66665 C3M6OK 155539896 IC50 = 14700 nM T66665 CD6SZ8 155540325 IC50 = 1210 nM T66665 C5R1KH 155542501 IC50 = 710 nM T66665 C06ILW 155542709 IC50 = 220 nM T66665 CJ6CD8 155542855 IC50 = 230 nM T66665 CNU2C0 155544451 IC50 = 1150 nM T66665 CEZ3U5 155544780 IC50 = 64.9 nM T66665 C53BXM 155545107 IC50 = 44500 nM T66665 CPQV84 155545220 IC50 = 190 nM T66665 C73WZV 155545478 IC50 > 500000 nM T66665 CK3EW2 155545512 IC50 = 52970 nM T66665 CB9V4N 155545715 IC50 = 103.17 nM T66665 C19VEP 155545723 IC50 = 300 nM T66665 CTQ1N5 155545760 IC50 = 190 nM T66665 CS3QE6 155545912 IC50 = 250 nM T66665 C30NDT 155546179 IC50 = 19.87 nM T66665 CF93IH 155546386 IC50 = 240 nM T66665 C02VES 155546488 IC50 = 9840 nM T66665 C08YIN 155547155 IC50 = 11 nM T66665 CM67HN 155547227 IC50 = 850 nM T66665 CPF8U1 155547250 IC50 = 380 nM T66665 CVP4G7 155547475 IC50 = 34.21 nM T66665 CS9TE8 155547623 IC50 = 450 nM T66665 CFR63D 155547749 IC50 = 170 nM T66665 CEV12A 155547825 IC50 = 5000 nM T66665 C76HDR 155547843 IC50 = 20 nM T66665 CJW4H5 155548487 IC50 = 10000 nM T66665 C4CY2L 155548534 IC50 = 43900 nM T66665 C7IES3 155548701 IC50 = 42700 nM T66665 CV6P2U 155549134 IC50 = 70000 nM T66665 C2RB6X 155549809 IC50 = 880 nM T66665 CK65AT 155550206 IC50 = 930 nM T66665 C3UBY1 155551683 IC50 = 130 nM T66665 CIXT57 155551691 IC50 = 7640 nM T66665 CC90IJ 155551771 IC50 = 110 nM T66665 CYDP17 155551847 IC50 = 38.73 nM T66665 CZO59G 155552038 IC50 = 44900 nM T66665 CH6E5X 155552439 IC50 = 260 nM T66665 CH3NT4 155552664 IC50 = 400 nM T66665 CJ3H8K 155552805 IC50 = 390 nM T66665 C9ZF0A 155552862 IC50 > 50000 nM T66665 CG1U2I 155553094 IC50 = 3990 nM T66665 C0BHJ2 155553248 IC50 = 2010 nM T66665 CYG31B 155553429 IC50 = 52.34 nM T66665 C3CG7H 155553481 IC50 = 7140 nM T66665 C7BM0W 155553539 IC50 = 11640 nM T66665 CND9J8 155553598 IC50 = 53900 nM T66665 CPZ0C9 155554102 IC50 = 100 nM T66665 CB18OG 155554424 IC50 = 640 nM T66665 CW9YD6 155554611 IC50 > 50000 nM T66665 CBD7W9 155555889 IC50 = 230 nM T66665 CM8B6E 155556262 IC50 = 660000 nM T66665 C37JXS 155556771 IC50 = 10100 nM T66665 C1HSK4 155557372 IC50 = 6220 nM T66665 CHGI70 155557383 IC50 = 46400 nM T66665 C9XRB6 155557877 IC50 = 670 nM T66665 CS96MZ 155557974 IC50 = 99000 nM T66665 CCV8M6 155558071 IC50 = 44900 nM T66665 CERZ85 155558072 IC50 = 720 nM T66665 CY3U6N 155558126 IC50 = 100 nM T66665 C4V6GB 155558213 IC50 = 9250 nM T66665 CHI7P2 155558802 IC50 = 460 nM T66665 CAX70V 155559496 IC50 = 3000 nM T66665 CVGD95 155559759 IC50 = 58.04 nM T66665 CF4W8Y 155559976 IC50 = 134.58 nM T66665 CMH04B 155560214 IC50 > 50000 nM T66665 CK9PR5 155560364 IC50 = 380 nM T66665 CT9W5F 155560713 IC50 = 350 nM T66665 CGO1Y6 155561686 IC50 > 50000 nM T66665 C50XAB 155562173 IC50 = 390 nM T66665 C2KMB7 155562273 IC50 = 560 nM T66665 C5ZBY8 155562605 IC50 = 430 nM T66665 CGD15R 155562754 IC50 = 270 nM T66665 C13BZU 155563007 IC50 = 430 nM T66665 C48GFH 155563162 IC50 = 210 nM T66665 CP8BG6 155563791 IC50 = 290 nM T66665 CX12MT 155563845 IC50 = 36.54 nM T66665 C53AWR 155563991 IC50 = 43.74 nM T66665 CV4I2Q 155564403 IC50 = 10330 nM T66665 CF7G4U 155565228 IC50 = 56100 nM T66665 C89DPY 155565424 IC50 = 110 nM T66665 C79ZDF 155566047 IC50 = 330 nM T66665 C28TBL 155567336 IC50 = 39.14 nM T66665 C9HJD2 155567394 IC50 = 24000 nM T66665 COC6J1 155567620 IC50 = 100 nM T66665 C93HQW 155567629 IC50 = 4500 nM T66665 CQK25N 155568033 IC50 > 100000 nM T66665 C3MN9X 155568608 IC50 = 31.91 nM T66665 CU3F4D 155568632 IC50 = 310 nM T66665 C70ZUA 155569262 IC50 = 13490 nM T66665 CR2S0C 108068 IC50 = 800 nM T66665 CC35YL 11335338 IC50 = 20 nM T66665 CL4VS1 118222242 IC50 = 14 nM T66665 CQF61C 118720946 IC50 = 9 nM T66665 D00AII 5281727 IC50 = 820 nM T66665 D00MXS 5281703 IC50 = 46000 nM T66665 D00RCV 9813643 IC50 = 3000 nM T66665 D00RIX 5280443 IC50 = 8000 nM T66665 D00VHS 136036233 IC50 > 50000 nM T66665 D00XIX 44564003 IC50 > 50000 nM T66665 D01BZE 73659 IC50 > 40000 nM T66665 D01EWD 9944615 IC50 = 12000 nM T66665 D01MFK 9906892 IC50 = 40 nM T66665 D01PBO 44423052 IC50 = 73900 nM T66665 D01SNR 208910 IC50 = 140 nM T66665 D01UYI 5281607 IC50 = 25500 nM T66665 D01VRB 44564456 IC50 = 4000 nM T66665 D01WLL 11460185 IC50 = 1190 nM T66665 D02CCB 23627032 IC50 = 1330 nM T66665 D02FEF 404378 IC50 = 5450 nM T66665 D02FGY 44434501 IC50 = 2400 nM T66665 D02GZX 9817355 IC50 = 330 nM T66665 D02PLG 44564508 IC50 = 20000 nM T66665 D02VLR 2211 IC50 = 800 nM T66665 D02XEX 11168203 IC50 > 40000 nM T66665 D03FXI 564225 IC50 = 3000 nM T66665 D03NMM 46843035 IC50 > 100000 nM T66665 D03TLR 44564454 IC50 > 50000 nM T66665 D03VUQ 404202 IC50 = 3420 nM T66665 D04JZY 46855201 IC50 = 8950 nM T66665 D04KAM 10220627 IC50 = 3500 nM T66665 D04YPP 9991673 IC50 = 2490 nM T66665 D05IWY 5464078 IC50 = 2000 nM T66665 D05JRZ 67316 IC50 = 8890 nM T66665 D05QOR 5280460 IC50 > 100000 nM T66665 D06DRL 44475843 IC50 = 2690 nM T66665 D06TPF 1057 IC50 = 144000 nM T66665 D06TXM 24816385 IC50 > 10 nM T66665 D06WML 10377376 IC50 = 1490 nM T66665 D06YGF 5281787 IC50 = 82000 nM T66665 D06ZRX 5281717 IC50 = 109000 nM T66665 D07LUJ 64945 IC50 > 40000 nM T66665 D07OAV 44424411 IC50 > 100000 nM T66665 D07QIU 625902 IC50 = 9880 nM T66665 D07STC 44434500 IC50 = 6200 nM T66665 D08QAH 44336344 IC50 = 2400 nM T66665 D08RCQ 44564416 IC50 > 50000 nM T66665 D09DMR 44456679 IC50 = 3110 nM T66665 D09VYW 9847548 IC50 > 40000 nM T66665 D09XCX 5694 IC50 > 10 nM T66665 D0BO9W 11150126 IC50 = 14110 nM T66665 D0C1GO 1396 IC50 = 50 nM T66665 D0CW3A 46855054 IC50 = 7530 nM T66665 D0D0JE 24884690 IC50 = 8000 nM T66665 D0E0RW 69894 IC50 > 100000 nM T66665 D0EI8V 45268661 IC50 = 12 nM T66665 D0F0JU 44564415 IC50 = 800 nM T66665 D0F3UR 690836 IC50 = 4940 nM T66665 D0F6CD 5202 IC50 > 400000 nM T66665 D0F9RO 6918774 IC50 > 40000 nM T66665 D0FQ3N 5748382 IC50 = 1890 nM T66665 D0G3TK 5280863 IC50 > 100000 nM T66665 D0G7RA 44564004 IC50 > 50000 nM T66665 D0I9AT 73549 IC50 = 64 nM T66665 D0J1AW 405560 IC50 = 2780 nM T66665 D0J7YE 17164245 IC50 = 107000 nM T66665 D0JQ1T 44336354 IC50 = 190 nM T66665 D0JT8Y 21177358 IC50 = 6750 nM T66665 D0K4QW 44219619 IC50 = 7700 nM T66665 D0L6TP 11277773 IC50 > 100000 nM T66665 D0LC7K 119034 IC50 > 40000 nM T66665 D0LJ7R 15345559 IC50 = 460 nM T66665 D0M5MI 4306515 IC50 > 3300 nM T66665 D0M7EI 9837624 IC50 = 5000 nM T66665 D0M9RL 44336367 IC50 = 150 nM T66665 D0N7OP 44424412 IC50 = 62300 nM T66665 D0N7XM 24992964 IC50 > 100000 nM T66665 D0NH1E 1383884 IC50 > 100000 nM T66665 D0O8XG 9965111 IC50 = 6500 nM T66665 D0O9NE 5388063 IC50 = 1667 nM T66665 D0OX0B 44424402 IC50 = 660 nM T66665 D0PJ3M 637511 IC50 = 245000 nM T66665 D0PQ3Q 44564458 IC50 > 50000 nM T66665 D0QV6M 4292 IC50 = 60 nM T66665 D0S2II 308405 IC50 = 2870 nM T66665 D0S7LD 5326145 IC50 = 2990 nM T66665 D0SJ2Q 10494 IC50 > 40000 nM T66665 D0T2SD 21862824 IC50 = 4620 nM T66665 D0T4VL 9908776 IC50 = 93300 nM T66665 D0U0YE 14762941 IC50 = 47 nM T66665 D0U8IF 10114 IC50 > 40000 nM T66665 D0UH3D 49837499 IC50 = 14000 nM T66665 D0V3PG 128861 IC50 = 60000000 nM T66665 D0V7AA 9064 IC50 = 93300 nM T66665 D0V9EN 689043 IC50 = 129700 nM T66665 D0VF6F 10244543 IC50 = 37500 nM T66665 D0X4LI 13015959 IC50 = 1000 nM T66665 D0X6RO 404324 IC50 = 2220 nM T66665 D0X9VY 9965195 IC50 = 2000 nM T66665 D0Y1YR 442793 IC50 = 125000 nM T66665 D0Y9ZO 21862753 IC50 = 4380 nM T66665 D0YI3V 44336157 IC50 = 730 nM T66665 D0Z1WF 405489 IC50 = 14630 nM T66665 D0ZA6G 6323491 IC50 = 27 nM T66665 D0ZI8Y 44583799 IC50 = 2200 nM T67102 D07XHO 4413 IC50 > 1000000 nM T67102 D0A0OO 65016 IC50 = 15200 nM T67102 D0EV6T 54682461 Ki = 15000 nM T67102 D0A5SA 56591871 IC50 > 10000 nM T67102 D0CG8S 71305058 IC50 > 200000 nM T67102 D0D8II 513956 IC50 > 50000 nM T67102 D0FE7H 9876120 Ki = 0.07 nM T67102 D0H6AG 51003469 IC50 = 820 nM T67102 D0H7PW 638024 IC50 = 42300 nM T67102 D0N1BF 44251605 IC50 = 15700 nM T67102 D0R4KK 51352361 IC50 > 100000 nM T67102 D0U3EP 445154 IC50 = 138000 nM T67102 D0Y0EP 67979346 IC50 = 16100 nM T67102 D0Y5NA 118435360 IC50 > 95300 nM T67102 D0HM5J 118253852 IC50 > 20000 nM T67102 D00XRK 447617 IC50 > 31000 nM T67102 D01LNG 10201696 Ki = 1.29 nM T67102 D04ZIJ 5478883 IC50 = 0.0016 ug.mL-1 T67102 D07PSP 5479205 Ki > 1000 nM T67102 CAD6F5 44330836 Ki = 560 nM T67102 C3G6QJ 24051 IC50 = 1000 nM T67102 CZ0JE7 31222 IC50 = 2400 nM T67102 C7A9BK 65023 IC50 = 7500 nM T67102 C9ZTV0 77079 IC50 = 1000 nM T67102 CT9HP8 157824 IC50 = 550 nM T67102 CYJ72V 226139 IC50 = 1000 nM T67102 C6HBV9 444581 IC50 > 1300000 nM T67102 C2AX7O 445304 Ki > 2000 nM T67102 C6VC4K 445649 IC50 = 6 nM T67102 C8NGY9 448772 IC50 > 500000 nM T67102 CV2P5E 454914 Ki = 100 nM T67102 CV58GA 460197 IC50 = 35 nM T67102 C9QD2H 460207 IC50 = 110 nM T67102 C19EDU 460213 IC50 = 60 nM T67102 C0TN7S 460238 IC50 = 380 nM T67102 CAG9E8 460240 IC50 = 1800 nM T67102 C58KVI 460241 IC50 = 1000 nM T67102 CCU6P0 460242 IC50 > 10000 nM T67102 CZ0U9B 461281 IC50 > 10000 nM T67102 CJLM24 461282 IC50 > 10000 nM T67102 C8QY7D 461294 IC50 > 10000 nM T67102 C43OUC 467651 IC50 = 8200 nM T67102 C3QW5Y 636516 IC50 = 4.45 ug.mL-1 T67102 C20JZF 1898613 IC50 > 300000 nM T67102 C8AED5 2832201 IC50 = 1800 nM T67102 CVR7P3 3781218 IC50 = 1000 nM T67102 CE24HD 4385881 IC50 = 1200 nM T67102 CGSC72 5287532 Ki = 448 nM T67102 CO58XD 5311161 IC50 > 100000 nM T67102 C81PIJ 5494406 IC50 = 6000 nM T67102 CDG23K 5494410 IC50 = 56 nM T67102 CPS5Z7 6539218 Ki = 21 nM T67102 CV5K3I 6539219 Ki = 980 nM T67102 C7UR8H 6539220 Ki = 41 nM T67102 CYA9X5 6539221 Ki = 4.9 nM T67102 CY6M5W 6539222 Ki = 459 nM T67102 CEX3D8 6539224 Ki > 4000 nM T67102 C9DOI1 6539225 Ki = 140 nM T67102 CR7A3L 6539226 Ki = 265 nM T67102 C0H5ZW 6539227 Ki = 217 nM T67102 CUQ6T5 6539228 Ki = 623 nM T67102 C32QNI 6539229 Ki = 473 nM T67102 CZN02I 6539230 Ki = 41 nM T67102 CXPO09 6539231 Ki = 1807 nM T67102 C4GX1T 6539232 Ki > 4000 nM T67102 C2YKM3 6539233 Ki = 52 nM T67102 COLZ28 6539234 Ki = 100 nM T67102 CJ14EB 6539235 Ki = 35 nM T67102 CQ5O9H 6539236 Ki > 5900 nM T67102 CIY71M 6539237 Ki = 322 nM T67102 CIWC50 6539238 Ki > 5900 nM T67102 C9VQZ4 6539239 Ki > 5900 nM T67102 C4AXO5 6539241 Ki > 2000 nM T67102 CY8HL5 6539242 Ki > 2000 nM T67102 CA78BY 6539243 Ki > 2000 nM T67102 CB2O4C 6539244 Ki > 2000 nM T67102 CEX54J 6539245 Ki > 2000 nM T67102 C61TOP 6539246 Ki > 2000 nM T67102 C01MAJ 6539247 Ki > 200 nM T67102 CV7NB4 6539248 Ki > 2000 nM T67102 CMHE43 6539249 Ki > 2000 nM T67102 CQO6I0 6539250 Ki > 2000 nM T67102 CHC57F 6539251 Ki > 2000 nM T67102 CT30RS 6539252 Ki > 2000 nM T67102 CNZ8E9 6539253 Ki > 2000 nM T67102 CV9Q8Z 6539254 Ki > 2000 nM T67102 C3VB5A 6539255 Ki > 2000 nM T67102 C6H5IQ 6539256 Ki > 2000 nM T67102 CF30BP 6539257 Ki = 30 nM T67102 CZ40TI 6539258 Ki > 2000 nM T67102 CQLC81 6539259 Ki = 320 nM T67102 CMNF51 6539260 Ki = 63 nM T67102 C3WI4Y 6539261 Ki > 2000 nM T67102 CE51XA 6539262 Ki > 2800 nM T67102 CN6OX1 6539263 Ki > 2000 nM T67102 CB89QP 6539264 Ki > 2800 nM T67102 CB14ZY 6539265 Ki > 2000 nM T67102 CBF54P 6539266 Ki > 2000 nM T67102 CM6X7H 6539267 Ki > 2000 nM T67102 C6RQ9Z 6539268 Ki ~ 1700 nM T67102 C0Y9GC 6539269 Ki ~ 1000 nM T67102 CWIJ07 6539270 Ki ~ 1700 nM T67102 CSD6R5 6539271 Ki > 2000 nM T67102 CWR7C9 6539272 Ki = 1700 nM T67102 CXT20F 6539273 Ki = 1900 nM T67102 CURY46 6539274 Ki = 1600 nM T67102 CLE4I2 6539275 Ki > 2000 nM T67102 C1SUG3 6539276 Ki > 2000 nM T67102 CV2JK1 6539277 Ki > 2000 nM T67102 CRS54N 6540293 Ki = 131 nM T67102 C3OD0J 6918853 IC50 = 70 nM T67102 CR59LJ 9547928 IC50 = 11 nM T67102 CPCN93 9547929 IC50 = 10 nM T67102 C2M4ZF 9801811 IC50 = 9400 nM T67102 COBW38 9821383 IC50 > 100000 nM T67102 CKP0I3 9830952 Ki = 1.3 nM T67102 C7Z8UC 9831520 Ki = 15 nM T67102 CX0B5L 9853618 IC50 > 100000 nM T67102 C35UMF 9890209 IC50 = 6.41 ug.mL-1 T67102 C0HM2T 9895330 Ki = 5.8 nM T67102 CLF04H 9938431 IC50 = 2950 nM T67102 CW67YS 9939419 IC50 = 630 nM T67102 CF7D2T 9960476 Ki = 9.8 nM T67102 C60RLE 9983009 IC50 = 210 nM T67102 C2P3DU 9983140 IC50 = 780 nM T67102 CIBZ30 9984485 IC50 = 18620 nM T67102 C93KNF 9986236 IC50 = 1020 nM T67102 CHG57R 9986500 IC50 = 1090 nM T67102 C17HZK 10005121 IC50 = 230 nM T67102 CN92WM 10005768 IC50 = 210 nM T67102 C8XV3Y 10008157 IC50 = 5750 nM T67102 CJ8B0Q 10028131 IC50 = 940 nM T67102 CO7A2D 10033021 Ki = 4.3 nM T67102 CEQP27 10049905 IC50 = 12 nM T67102 CN2J9E 10054920 IC50 = 350 nM T67102 CY9SK0 10073810 IC50 = 10960 nM T67102 CEFK38 10077756 IC50 = 5145 nM T67102 CAKR94 10077830 IC50 = 350 nM T67102 CJ4TR1 10078059 IC50 = 680 nM T67102 CSA7C0 10098656 IC50 = 193 nM T67102 C0LOV8 10100288 IC50 = 450 nM T67102 CK51FX 10100482 IC50 = 110 nM T67102 C9F4ER 10120976 IC50 = 150 nM T67102 CE46MS 10146435 IC50 = 67 nM T67102 C2UNQ0 10258545 IC50 = 405 nM T67102 CB60PQ 10258985 IC50 = 170 nM T67102 CJZ98B 10324013 IC50 = 970 nM T67102 C3QN7I 10326962 IC50 = 520 nM T67102 CM46XO 10327211 IC50 = 430 nM T67102 C9Z2BY 10327349 Ki = 71 nM T67102 CML3K5 10348155 IC50 = 5010 nM T67102 CN89XA 10369729 IC50 = 9770 nM T67102 CQ0Y7C 10371570 IC50 = 280 nM T67102 CIA94Y 10371854 IC50 = 600 nM T67102 CZ5J7R 10391277 IC50 = 19050 nM T67102 C5C0JY 10393370 Ki = 200 nM T67102 C69KGX 10394329 Ki = 2.5 nM T67102 CZK1G9 10413386 IC50 = 9550 nM T67102 CYL37G 10415909 IC50 = 3550 nM T67102 CEYO32 10416248 IC50 = 660 nM T67102 CTN8C4 10417402 IC50 = 250 nM T67102 C8F3EC 10438938 IC50 = 2140 nM T67102 CJU80M 10439665 IC50 = 350 nM T67102 CZ6GK9 10461757 IC50 = 640 nM T67102 CL27YN 10462501 Ki = 58 nM T67102 CYE70D 10483879 IC50 = 207 nM T67102 C74JHX 10483887 IC50 = 400 nM T67102 CN68BR 10484078 IC50 = 980 nM T67102 C21ANW 10485108 Ki = 5300 nM T67102 CKXB12 10508444 Ki = 1.9 nM T67102 C1GYV7 10931081 IC50 = 251 nM T67102 CV01KW 11106059 IC50 = 1000 nM T67102 C3RQ9I 11157167 IC50 = 2110 nM T67102 C6HBJ0 11168125 IC50 = 75500 nM T67102 CZ40LC 11169672 IC50 < 10 nM T67102 CEX8G1 11178891 IC50 = 6610 nM T67102 C06BES 11192316 IC50 = 570 nM T67102 CQ71PI 11193205 IC50 = 28 nM T67102 CN0F8E 11199915 IC50 > 100000 nM T67102 C0J2NU 11204230 Ki > 5900 nM T67102 C9LK4F 11204313 IC50 = 25 nM T67102 CN8IX6 11215318 IC50 = 14120 nM T67102 CY7IP9 11215540 IC50 = 1000 nM T67102 COWF09 11215541 IC50 = 660 nM T67102 CEDP95 11215989 Ki = 1440 nM T67102 CJHM10 11227304 IC50 = 150 nM T67102 CENB36 11227366 Ki = 685 nM T67102 CH81IQ 11227430 IC50 = 780 nM T67102 CH3RF8 11227663 IC50 < 10 nM T67102 CEW9L6 11228293 Ki = 540 nM T67102 C4HXV1 11232421 Ki = 740 nM T67102 CU0C8V 11238286 IC50 = 6790 nM T67102 CE1B6S 11239445 Ki = 2701 nM T67102 CX30NP 11249866 Ki = 3600 nM T67102 CG87MJ 11250223 IC50 = 300 nM T67102 CZ4X0A 11250844 Ki = 1730 nM T67102 C9L7RA 11262610 IC50 = 130 nM T67102 C8PHK2 11273154 Ki = 481 nM T67102 C9W2NY 11274374 Ki = 4300 nM T67102 CR3YE1 11284734 IC50 = 90 nM T67102 C2C4XA 11285489 Ki = 2.5 nM T67102 C4BHV0 11285517 Ki = 1.6 nM T67102 C98FEY 11285691 Ki > 6000 nM T67102 CU80VL 11290116 IC50 = 60000 nM T67102 C9E0FG 11295146 IC50 = 34590 nM T67102 C4WK2S 11295726 IC50 = 36310 nM T67102 C5BO7P 11296167 Ki = 241 nM T67102 C7FKT1 11296858 IC50 = 1260 nM T67102 CNS4B0 11296859 IC50 = 1259 nM T67102 CX0GT9 11307634 IC50 = 60 nM T67102 C2QK0E 11308017 Ki = 1880 nM T67102 CM3G0J 11308211 IC50 = 660 nM T67102 CY5GU3 11308212 IC50 = 1000 nM T67102 CV8J9H 11308746 IC50 = 60 nM T67102 CM6Y4N 11319368 IC50 = 430 nM T67102 CVDC34 11329962 IC50 = 5430 nM T67102 C0SY2J 11330997 IC50 = 98 nM T67102 CL0P2H 11342148 IC50 = 1190 nM T67102 CY78LG 11377351 IC50 = 5010 nM T67102 C1RG5P 11399816 Ki = 3.9 nM T67102 C6UT8Z 11399839 Ki = 3.2 nM T67102 CC72ZR 11406807 IC50 = 60 nM T67102 CSJD04 11410402 Ki = 4940 nM T67102 CJS69P 11410845 IC50 = 1500 nM T67102 CEM8Q5 11444313 IC50 = 7930 nM T67102 C3ZI7O 11444912 IC50 = 1620 nM T67102 CR4F1K 11456236 IC50 = 17180 nM T67102 CLK8V9 11467715 IC50 = 1000 nM T67102 C0OPF5 11467778 IC50 = 2960 nM T67102 CUVZ93 11468096 IC50 = 1230 nM T67102 CH2Y7V 11478322 IC50 = 19540 nM T67102 CRZ86I 11498384 Ki = 304 nM T67102 C2RXZ9 11499243 Ki = 30800 nM T67102 C9YKP7 11505733 Ki > 6000 nM T67102 CJ9NL1 11505900 Ki > 6000 nM T67102 C2LD3N 11510567 IC50 = 8180 nM T67102 CK0L9W 11510740 IC50 = 78700 nM T67102 C1VEC2 11513333 Ki > 6000 nM T67102 C8P5JQ 11513415 Ki > 6000 nM T67102 C3P6ZU 11516577 IC50 = 12500 nM T67102 CYIV63 11517020 IC50 = 6700 nM T67102 CW68BJ 11518143 IC50 > 30000 nM T67102 C5XB3T 11520033 Ki = 32 nM T67102 CF2JU9 11520423 Ki > 6000 nM T67102 CK2JD4 11525068 IC50 = 4250 nM T67102 C6U9JR 11527693 Ki > 6000 nM T67102 C2VN5E 11531131 IC50 = 21440 nM T67102 CIK75C 11532248 IC50 = 3510 nM T67102 CPK79W 11532880 IC50 = 6900 nM T67102 C5QB4G 11533200 IC50 = 476 nM T67102 CKU80T 11534178 Ki > 6000 nM T67102 CKY5C8 11534582 Ki > 6000 nM T67102 CS0H9X 11534953 Ki > 6000 nM T67102 C2W8MQ 11538592 IC50 = 2470 nM T67102 CT50OI 11539235 IC50 = 12200 nM T67102 C6CVW2 11539562 IC50 = 2330 nM T67102 CR93VK 11539712 IC50 = 36200 nM T67102 C02DGS 11541427 Ki > 6000 nM T67102 C8SFN6 11541810 Ki > 6000 nM T67102 C2IL9N 11543843 IC50 > 100000 nM T67102 C0KY4O 11545958 IC50 = 6280 nM T67102 CYEL51 11553053 IC50 = 9200 nM T67102 CSL71C 11553983 IC50 = 1870 nM T67102 CE9ZI8 11556254 Ki = 36 nM T67102 CZ07VP 11560610 IC50 = 2190 nM T67102 CB59KM 11564069 Ki = 1200 nM T67102 C8OUD5 11576737 IC50 = 144 nM T67102 CR8AL4 11582999 Ki = 19300 nM T67102 CE6CH3 11583947 IC50 = 18900 nM T67102 CA29QF 11589453 IC50 = 23100 nM T67102 C9FI7P 11590166 IC50 = 12500 nM T67102 C1A7SE 11596660 IC50 = 43600 nM T67102 C0EOP4 11604171 IC50 = 24700 nM T67102 CV30CG 11604834 IC50 = 73500 nM T67102 CZ1V8Y 11606008 IC50 = 2100 nM T67102 C8RPH4 11607313 Ki > 6000 nM T67102 CT97EJ 11611402 IC50 = 10300 nM T67102 CL9V5H 11611694 IC50 = 12200 nM T67102 C1PSL5 11614083 Ki = 291 nM T67102 C7XU9H 11614671 Ki > 6000 nM T67102 CFU9Q3 11618427 IC50 = 24900 nM T67102 CMW5Y1 11618935 IC50 = 54100 nM T67102 CAP36L 11619283 IC50 = 6450 nM T67102 C7ZWK0 11620576 IC50 = 470 nM T67102 CSR87I 11629093 Ki > 6000 nM T67102 C3LW2D 11632240 IC50 = 11000 nM T67102 CUD76B 11632510 IC50 = 5200 nM T67102 C78KYL 11633041 IC50 = 16500 nM T67102 C2QC4B 11633904 IC50 = 8300 nM T67102 CN9AO7 11636216 Ki > 6000 nM T67102 COC2F0 11639859 IC50 = 7300 nM T67102 CED2Y7 11640634 IC50 = 19400 nM T67102 C8DZG9 11647909 IC50 = 16440 nM T67102 C6MH7K 11648455 IC50 = 18100 nM T67102 C0UXN3 11654224 IC50 = 10900 nM T67102 CSKL32 11654876 IC50 = 10100 nM T67102 CT13BA 11655737 IC50 = 56900 nM T67102 CEU6R3 11655813 IC50 = 3010 nM T67102 CA45GE 11657449 Ki > 6000 nM T67102 CHXL54 11664893 Ki > 6000 nM T67102 C4PXM5 11668120 IC50 = 23920 nM T67102 C14JYI 11668187 IC50 = 14300 nM T67102 CY47BE 11683112 IC50 = 93700 nM T67102 CXN6V9 11685086 Ki > 6000 nM T67102 CB2GA5 11697219 IC50 = 44300 nM T67102 CU57OC 11705307 IC50 > 100000 nM T67102 CWTA90 11707562 Ki > 6000 nM T67102 CK73DU 11710655 IC50 = 52500 nM T67102 CBJ08S 11711024 IC50 = 69500 nM T67102 CIDF31 11721953 Ki = 800 nM T67102 CHEI17 11754571 IC50 = 24 nM T67102 CGE50S 11757267 Ki = 79700 nM T67102 CH1Y8K 11764107 Ki = 0.7 nM T67102 CF1CZ0 11765081 IC50 = 580 nM T67102 CN7AX1 11765192 IC50 = 250 nM T67102 CJN0K9 11765311 IC50 = 550 nM T67102 CQZR02 11765842 Ki = 5.2 nM T67102 CF1RT6 11785879 IC50 = 58880 nM T67102 CG2HY0 11785880 IC50 = 58880 nM T67102 CVQ7O2 11786748 IC50 = 60 nM T67102 CD1N7A 11787369 Ki = 32 nM T67102 CR5M7I 11845063 IC50 = 9000 nM T67102 CV8XS9 11845069 IC50 > 10000 nM T67102 CEK56D 11845403 IC50 > 10000 nM T67102 C8H1ES 11845584 IC50 = 6900 nM T67102 C0W1KA 11845953 IC50 > 10000 nM T67102 CJ34FE 11845955 IC50 > 10000 nM T67102 CX34FU 11846304 IC50 = 180 nM T67102 CUON19 11846305 IC50 = 20 nM T67102 CI72TF 11846306 IC50 = 195 nM T67102 C38JYH 11846473 IC50 = 460 nM T67102 CICT21 11846474 IC50 = 9700 nM T67102 C8YEH5 11846475 IC50 = 1700 nM T67102 CKR6T3 11846476 IC50 = 3600 nM T67102 CHC79W 11846478 IC50 = 3900 nM T67102 CPO8E1 11846645 IC50 = 50 nM T67102 CG1UP6 11846815 IC50 = 1110 nM T67102 CE2OQ9 11846965 IC50 = 25 nM T67102 CR3G5X 11846966 IC50 = 190 nM T67102 C25PFL 11846967 IC50 = 1250 nM T67102 CU2TQ6 11846968 IC50 > 10000 nM T67102 CVQ9U5 11847590 IC50 = 200 nM T67102 CLP92O 11963435 IC50 > 30000 nM T67102 CGOD35 11990754 IC50 = 9400 nM T67102 CQ8SJ5 11990755 IC50 = 28500 nM T67102 CE25DJ 13851954 IC50 = 1700 nM T67102 CE29TK 14887165 IC50 = 600 nM T67102 CJO10Z 14887166 IC50 > 10000 nM T67102 C02NGW 14887167 IC50 > 10000 nM T67102 CJ8R0O 14887174 IC50 = 175 nM T67102 CHIC86 14887175 IC50 = 250 nM T67102 C56EWA 14887177 IC50 = 115 nM T67102 C2LRD8 14887179 IC50 = 280 nM T67102 CT4V6C 14887181 IC50 = 150 nM T67102 C4UA0C 14887183 IC50 = 100 nM T67102 C6JF8N 14887185 IC50 = 500 nM T67102 CAKS64 14887194 IC50 ~ 5000 nM T67102 CE12CX 15018069 Ki = 0.8 nM T67102 CI41XT 15126555 Ki = 0.4 nM T67102 C9KCN0 15546672 Ki = 231 nM T67102 CRNW82 15546675 Ki = 3 nM T67102 CR4G6J 15949919 IC50 = 22000 nM T67102 CQ3GX2 15950003 IC50 = 1470 nM T67102 C3CI9Z 15950004 IC50 = 1910 nM T67102 C2BQ4V 15950005 IC50 = 11300 nM T67102 C6QD9U 15950006 IC50 = 11900 nM T67102 CW4US1 15950085 IC50 = 38600 nM T67102 CZM1C9 15950086 IC50 = 4030 nM T67102 C8Y6UT 15950518 IC50 = 31600 nM T67102 CAPV27 15950520 IC50 = 46800 nM T67102 C0J9PD 15951416 IC50 = 30000 nM T67102 CSQ3X1 15951420 IC50 = 20800 nM T67102 C8IZR0 15951484 IC50 = 34100 nM T67102 CB1G7D 15951486 IC50 = 14100 nM T67102 CNPJ39 15951487 IC50 = 24200 nM T67102 CE67NK 15951489 IC50 = 12200 nM T67102 CW6S0H 15981486 IC50 = 2653 nM T67102 C0QAD8 16050550 IC50 = 15320 nM T67102 C1CEU6 16050551 IC50 = 11530 nM T67102 CX8O6Q 16050552 IC50 = 8400 nM T67102 CYQ7X3 16050553 IC50 = 14100 nM T67102 C2WR8B 16050640 IC50 = 27280 nM T67102 CF5EC0 16050641 IC50 = 36600 nM T67102 C4DO8C 16050931 IC50 = 24000 nM T67102 C0Q2MC 16051586 IC50 = 17100 nM T67102 CIV72W 16086657 IC50 = 2700 nM T67102 CAY1B5 16090342 IC50 = 25000 nM T67102 CP5G7V 16090348 IC50 = 5900 nM T67102 C2HMT5 16113206 IC50 = 2980 nM T67102 CX39UL 16113753 IC50 = 53000 nM T67102 CJDF09 16129583 IC50 = 2400 nM T67102 CL26VD 16659019 Ki = 245 nM T67102 CGU76F 16659022 Ki = 490 nM T67102 C73FHN 16659067 Ki = 483 nM T67102 C01GFZ 16659107 Ki = 633 nM T67102 CVM2G8 16725331 Ki = 510 nM T67102 CRW5Q2 16730753 IC50 = 28 nM T67102 CI7Z6F 16741239 IC50 = 110 nM T67102 CMXW48 21085652 IC50 = 3600 nM T67102 CU2E5X 21087080 IC50 > 20000 nM T67102 C9NZ6L 21191206 IC50 = 33000 nM T67102 CAX1F4 21191209 IC50 = 17600 nM T67102 C2RCK6 21191217 IC50 = 640 nM T67102 CBV5Q6 21191229 IC50 = 2980 nM T67102 C9OWG1 21191244 IC50 = 1310 nM T67102 CGL93J 21191246 IC50 = 14100 nM T67102 CZOU03 21191268 IC50 = 2560 nM T67102 CZIS68 21191280 IC50 = 48400 nM T67102 CV1YP5 21191290 IC50 = 1860 nM T67102 C0VRG5 21191297 IC50 = 780 nM T67102 CMXJ30 23625795 IC50 > 10000 nM T67102 C0T8KQ 23647294 IC50 = 150 nM T67102 C17VPL 23647295 IC50 = 260 nM T67102 CG46BK 23647296 IC50 = 190 nM T67102 CK40YS 23657802 IC50 = 2510 nM T67102 C4BR2E 23657804 IC50 = 600 nM T67102 CEI3N7 24794397 IC50 = 3900 nM T67102 C2VT1S 24801864 Ki = 195 nM T67102 CT96WK 24801865 Ki = 80 nM T67102 CJUX10 24808497 Ki = 47 nM T67102 CE05DA 24877512 IC50 = 1800 nM T67102 CB9DT6 24877514 IC50 = 1900 nM T67102 C3EHC6 24877515 IC50 = 1700 nM T67102 C1ILH2 24877517 IC50 = 2400 nM T67102 CV7FB1 24877625 IC50 = 1200 nM T67102 CA37MN 24877744 IC50 = 5400 nM T67102 C4SZA8 24877746 IC50 = 1900 nM T67102 CUW1D7 24877749 IC50 = 2300 nM T67102 CFJ87K 24877750 IC50 = 2000 nM T67102 C9IKJ2 24877858 IC50 = 2400 nM T67102 CWM1Q4 24878892 IC50 = 26300 nM T67102 CTO0H5 24878893 IC50 = 26300 nM T67102 CKWX57 24878894 IC50 = 5250 nM T67102 CF0Q3S 24878945 IC50 = 30200 nM T67102 C09LYN 24878946 IC50 = 30200 nM T67102 CI54AT 24878947 IC50 > 100000 nM T67102 C8LQ5C 24882338 IC50 = 2695 nM T67102 CMJK34 24882477 IC50 = 380 nM T67102 C32SYP 24950594 IC50 = 2400 nM T67102 C6WD3C 24969880 IC50 = 41 nM T67102 C50CQN 25066229 IC50 = 9 nM T67102 CT9MX8 25066444 Ki = 66 nM T67102 CO7MQ2 25069561 IC50 = 3400 nM T67102 C8ANG7 25070193 IC50 = 1800 nM T67102 C0T8LP 25070195 IC50 = 22500 nM T67102 CM37LQ 25072736 IC50 = 2000 nM T67102 C0UO6V 25073049 IC50 = 2120 nM T67102 CL3QK6 25096211 IC50 = 59 nM T67102 C2UWA1 25096462 Ki = 3.3 nM T67102 CZV97Q 25096707 IC50 = 120 nM T67102 C3H6BD 25110732 Ki = 630 nM T67102 C93HLR 25113163 Ki = 780 nM T67102 C4E9MK 25120557 IC50 > 25000 nM T67102 CU7P0M 25120899 IC50 = 599 nM T67102 C4KM6T 25121609 IC50 = 1380 nM T67102 CNTF43 25127621 IC50 = 3750 nM T67102 C4E0MJ 25127622 IC50 = 1500 nM T67102 CWF5Z3 25143506 IC50 > 30000 nM T67102 CEUT61 25156748 Ki = 61 nM T67102 C9WN6Q 25156749 Ki = 130 nM T67102 CG54TK 25157024 Ki = 240 nM T67102 CH8YV1 25157025 Ki = 3350 nM T67102 COK8S4 25163980 IC50 = 370 nM T67102 C6YWX8 25163981 IC50 > 10000 nM T67102 CKM2U5 25163982 IC50 = 1400 nM T67102 C3XDW1 25184934 IC50 = 11300 nM T67102 CS2MU5 25184935 IC50 = 33000 nM T67102 CXE56W 25184936 IC50 = 10800 nM T67102 CF91ST 25184937 IC50 = 10700 nM T67102 CSM9C5 25190481 IC50 = 34325 nM T67102 CU80RW 25190482 IC50 = 1750 nM T67102 CK48PJ 25190483 IC50 = 2940 nM T67102 CW6QJ1 25190484 IC50 = 2020 nM T67102 CKZ2Q7 25190485 IC50 = 8510 nM T67102 CWN51E 25190486 IC50 = 5890 nM T67102 C69RHT 25190487 IC50 = 4790 nM T67102 CT8N2P 25190488 IC50 = 25120 nM T67102 CJ6SA2 25190489 IC50 = 6170 nM T67102 CESB62 25190490 IC50 = 2570 nM T67102 CLS3O2 25190491 IC50 = 3090 nM T67102 CZY6C4 25190492 IC50 = 1070 nM T67102 C04QGB 25190493 IC50 = 56230 nM T67102 CF8U0N 25190494 IC50 = 6760 nM T67102 CX4PB5 25190495 IC50 = 2400 nM T67102 CKYP06 25190496 IC50 = 15140 nM T67102 CNXG37 25190497 IC50 > 100000 nM T67102 CTS92Q 25190499 IC50 = 6545 nM T67102 CY02QR 25190500 IC50 = 87100 nM T67102 CYN2X5 25195985 IC50 = 600 nM T67102 CZP06K 25195988 IC50 = 2220 nM T67102 COZ9A0 25196089 IC50 = 390 nM T67102 CGWR85 25196090 IC50 = 680 nM T67102 CU8ON3 25232084 Ki = 612 nM T67102 C40ITP 25232817 Ki = 520 nM T67102 CA9K0S 25232818 Ki = 290 nM T67102 C5G2BP 25232984 Ki = 320 nM T67102 CR9O7I 25232986 Ki = 590 nM T67102 CSO74W 25233156 Ki = 190 nM T67102 CI68AZ 25233160 Ki = 431 nM T67102 C6E5PM 25233329 Ki = 276 nM T67102 C9JEA2 25233330 Ki = 354 nM T67102 CFY28W 25233331 Ki = 450 nM T67102 C9XA8E 25233503 Ki = 417 nM T67102 C6CAS8 25233845 Ki = 1125 nM T67102 CMS9A5 25233846 Ki = 1302 nM T67102 C9H3IT 35756036 IC50 = 39200 nM T67102 CQH0F2 42636932 IC50 = 1 nM T67102 C7E0VB 44024156 IC50 = 14200 nM T67102 CD0BS4 44024183 IC50 = 31900 nM T67102 C3RO7F 44143253 IC50 = 1700 nM T67102 CXV1A7 44143258 IC50 = 4270 nM T67102 CWI68J 44143259 IC50 = 3720 nM T67102 CNQ97G 44143260 IC50 = 980 nM T67102 C95LPG 44143261 IC50 = 600 nM T67102 CV9K7F 44143262 IC50 = 53700 nM T67102 C0WRT2 44143263 IC50 = 13490 nM T67102 CWQ6L4 44143264 IC50 = 4070 nM T67102 CZ9MQ7 44143265 IC50 = 14130 nM T67102 C8EI0C 44143266 IC50 = 11220 nM T67102 CAJ0I2 44143267 IC50 = 3720 nM T67102 C7AH8B 44143268 IC50 = 15140 nM T67102 CFJ82W 44143269 IC50 = 14390 nM T67102 CQ34LK 44143270 IC50 = 23990 nM T67102 C7FQ8W 44143271 IC50 = 600 nM T67102 CCUX36 44143272 IC50 = 35480 nM T67102 CDR56H 44143274 IC50 = 1210 nM T67102 CNWC13 44143275 IC50 = 19950 nM T67102 C4C0WD 44143276 IC50 = 4100 nM T67102 C5SLK9 44143277 IC50 = 890 nM T67102 C39WZR 44143278 IC50 = 1070 nM T67102 CVF5L8 44143280 IC50 = 8150 nM T67102 CPX9B2 44143282 IC50 = 12300 nM T67102 C6CQM2 44143283 IC50 = 2160 nM T67102 CDEU24 44143285 IC50 = 15140 nM T67102 CD8WS6 44143286 IC50 = 2970 nM T67102 C7ZNM2 44193108 IC50 = 12700 nM T67102 C9D1YN 44193111 IC50 = 10700 nM T67102 CQ90YP 44193304 IC50 = 12600 nM T67102 CJ8DS1 44198935 IC50 > 3000000 nM T67102 C8Y9NQ 44219712 IC50 > 100000 nM T67102 C5S6QR 44253975 IC50 = 1620 nM T67102 CN9BZ7 44253976 IC50 = 7.3 nM T67102 C1XKV6 44280079 Ki > 100000 nM T67102 CC0UX3 44280080 Ki ~ 10000 nM T67102 CXS78Z 44280081 Ki = 73 nM T67102 CKWX45 44280100 Ki > 5000 nM T67102 C17TUV 44308538 IC50 = 6640 nM T67102 C8D9TW 44308540 IC50 = 9740 nM T67102 CZYU80 44308553 IC50 = 1460 nM T67102 C5VAQ1 44308713 IC50 = 3690 nM T67102 CYB5H2 44308714 IC50 = 2760 nM T67102 C0S8JQ 44308715 IC50 = 2940 nM T67102 CV5A3S 44308835 IC50 = 820 nM T67102 CKD6N0 44308859 IC50 = 5130 nM T67102 CXCU36 44308860 IC50 = 620 nM T67102 CX58CS 44308917 IC50 = 690 nM T67102 C1HC3E 44308918 IC50 = 7940 nM T67102 CR4X6W 44308938 IC50 = 7200 nM T67102 C70PTI 44314034 Ki = 700 nM T67102 CU9QX3 44314035 Ki = 1300 nM T67102 C80PUQ 44314036 Ki = 110 nM T67102 C7R6LH 44314039 Ki = 320 nM T67102 CK18PR 44314180 IC50 = 5500 nM T67102 CPY54X 44314225 Ki = 3900 nM T67102 C2KA5V 44314256 Ki = 50 nM T67102 COX2F9 44314257 IC50 = 500 nM T67102 CM8EQ3 44314285 Ki = 200 nM T67102 CP2TM3 44314353 Ki = 920 nM T67102 CMW07C 44314384 Ki = 560 nM T67102 CUC6H9 44318741 IC50 = 2000 nM T67102 CCH31R 44318753 IC50 = 1500 nM T67102 CD4B3K 44318906 IC50 = 460 nM T67102 CUJC86 44318922 IC50 > 7000 nM T67102 C7BQK5 44318932 IC50 = 1100 nM T67102 CV32IE 44318933 IC50 = 2000 nM T67102 C6JAW3 44318939 IC50 = 2500 nM T67102 CBLM04 44318945 IC50 = 5000 nM T67102 CA91GR 44318953 IC50 > 10000 nM T67102 CJI3V9 44318960 IC50 = 700 nM T67102 CIQ1B4 44318967 IC50 = 1300 nM T67102 CFTJ12 44318968 IC50 = 1600 nM T67102 CU1ZT5 44319013 IC50 = 1800 nM T67102 C63UXV 44319014 IC50 = 2200 nM T67102 CF7I3T 44319019 IC50 = 780 nM T67102 CN36LG 44319020 IC50 = 2800 nM T67102 CB7X3U 44319028 IC50 = 2700 nM T67102 CGT2W9 44319029 IC50 = 3800 nM T67102 CB4KA0 44319035 IC50 = 3200 nM T67102 C9L2MZ 44319074 IC50 = 3000 nM T67102 C0LGQ5 44319092 IC50 = 7200 nM T67102 C8OHW7 44319135 IC50 = 600 nM T67102 CVP5M7 44319136 IC50 = 490 nM T67102 C1HJ0F 44319190 IC50 = 2000 nM T67102 CHM3W8 44319202 IC50 > 10000 nM T67102 CJR6X5 44319203 IC50 > 10000 nM T67102 CNG75A 44319204 IC50 = 5500 nM T67102 CWRC78 44319209 IC50 = 1300 nM T67102 CW58RS 44319226 IC50 = 1500 nM T67102 C42CUA 44319227 IC50 = 2400 nM T67102 CK82OX 44319228 IC50 = 2000 nM T67102 CV79CS 44319386 IC50 = 1800 nM T67102 C1Y9OA 44319395 IC50 = 2500 nM T67102 C46APG 44319396 IC50 > 10000 nM T67102 CXN53H 44319411 IC50 > 10000 nM T67102 CS7XD5 44321765 Ki = 0.1 nM T67102 C2OFK8 44321766 Ki = 0.6 nM T67102 CZ45LH 44322035 Ki = 208 nM T67102 CQ09YG 44322074 Ki = 6.1 nM T67102 C3N9LQ 44322075 Ki = 15 nM T67102 CK0BQ2 44322083 Ki > 10000 nM T67102 CNT69K 44322084 Ki = 5.4 nM T67102 CN58AQ 44322086 Ki = 45 nM T67102 C1G0FY 44322087 Ki = 13 nM T67102 CILR20 44327511 Ki = 560 nM T67102 CQ0F2W 44327556 Ki = 320 nM T67102 CVAJ58 44327796 Ki = 50 nM T67102 C26ZNS 44327901 Ki = 200 nM T67102 CGJ9B1 44327927 Ki = 5500 nM T67102 C8JQ3R 44328032 Ki = 200 nM T67102 CUNS68 44328035 Ki = 2400 nM T67102 C3Q0UM 44328055 Ki = 1600 nM T67102 CKF62V 44328096 Ki = 1300 nM T67102 CVXC94 44328097 Ki = 110 nM T67102 C9PCO5 44328098 Ki = 920 nM T67102 CQGI84 44328099 Ki = 3900 nM T67102 CW9CZ3 44328100 Ki = 2100 nM T67102 CPF13H 44335353 IC50 = 2000 nM T67102 CPL8E9 44338421 Ki = 1800 nM T67102 CHKG96 44338599 Ki = 1100 nM T67102 CM8DR0 44338623 IC50 ~ 45000 nM T67102 CDK84O 44340607 IC50 > 10000 nM T67102 CY91SZ 44341490 Ki = 586 nM T67102 CWJ8T7 44342184 IC50 = 550 nM T67102 CL6I2E 44342257 IC50 = 110 nM T67102 C1VBW4 44342328 IC50 = 770 nM T67102 C8W2MR 44342329 Ki = 0.7 nM T67102 CP26NT 44342415 IC50 = 58000 nM T67102 CF3A4M 44343168 IC50 = 10000 nM T67102 CT0HM5 44368301 IC50 > 1000000 nM T67102 C3L4OX 44370362 IC50 = 12500 nM T67102 CK07AQ 44370533 Ki = 2200 nM T67102 CFB98M 44370558 Ki = 28000 nM T67102 CA2C1S 44370759 Ki = 12500 nM T67102 CM1HG2 44379569 Ki = 200 nM T67102 C3LA2W 44379720 Ki = 2 nM T67102 CMB9W5 44383534 IC50 = 135 nM T67102 CBRX02 44386708 IC50 > 10000 nM T67102 C4PW0V 44413924 IC50 = 910 nM T67102 CD62TC 44413943 IC50 = 110 nM T67102 CJV8O2 44413944 IC50 = 6000 nM T67102 CMC1X9 44415487 IC50 > 1000000 nM T67102 CR4OF3 44415504 IC50 > 1000000 nM T67102 CX0L6N 44415666 IC50 = 12290 nM T67102 C73IKD 44415697 IC50 = 8900 nM T67102 CP2S8E 44415718 IC50 = 231500 nM T67102 CH69JN 44415719 IC50 > 1000000 nM T67102 CL5V2I 44415741 IC50 = 4710 nM T67102 C5U6BK 44415757 IC50 > 1000000 nM T67102 CU92KH 44415803 IC50 = 140 nM T67102 CXC57A 44421346 IC50 = 7620 nM T67102 CBQ57P 44426031 IC50 = 450 nM T67102 C04GKL 44426032 IC50 = 2800 nM T67102 CBLF97 44426033 IC50 = 660 nM T67102 CZH59K 44426035 IC50 = 570 nM T67102 CPY4W3 44426036 IC50 > 20000 nM T67102 CVG7S6 44426039 IC50 > 20000 nM T67102 CJ2PI1 44426041 IC50 = 3600 nM T67102 C4OZ6F 44426043 IC50 = 1600 nM T67102 CP80YT 44426045 IC50 > 20000 nM T67102 C12NXL 44426048 IC50 = 3800 nM T67102 C25NTL 44426051 IC50 = 866 nM T67102 CU4B2Y 44441701 IC50 = 275000 nM T67102 C6QMY7 44441703 IC50 = 97000 nM T67102 C2JE8M 44441743 IC50 = 48000 nM T67102 C6G8VL 44445142 IC50 = 11202 nM T67102 C31TEH 44445143 IC50 = 6042 nM T67102 C97WEK 44445144 IC50 > 20000 nM T67102 C47PWX 44445145 IC50 = 6946 nM T67102 C7I0VE 44445146 IC50 = 7593 nM T67102 CDWQ62 44445147 IC50 > 20000 nM T67102 CX50FP 44445148 IC50 = 10986 nM T67102 CX6IA7 44445149 IC50 = 9669 nM T67102 C4FRC0 44445150 IC50 > 20000 nM T67102 CC3Z0V 44445151 IC50 > 20000 nM T67102 C1XRF3 44445152 IC50 = 2116 nM T67102 CXH12K 44445153 IC50 = 4900 nM T67102 CTH2D6 44445154 IC50 = 11700 nM T67102 CFQ21V 44445155 IC50 = 4880 nM T67102 C68VFD 44446196 IC50 = 7700 nM T67102 C4S1CA 44446197 IC50 = 2400 nM T67102 C7K1RZ 44446198 IC50 = 1550 nM T67102 C5CS2Z 44446199 IC50 = 12020 nM T67102 CZO7A4 44446200 IC50 = 1095 nM T67102 CJVG08 44446201 IC50 = 10720 nM T67102 CF7RP8 44446202 IC50 = 22325 nM T67102 CU54SK 44446203 IC50 = 930 nM T67102 CJ3BD7 44446204 IC50 = 4680 nM T67102 CJW16S 44446205 IC50 = 1780 nM T67102 CSPE84 44446206 IC50 = 5250 nM T67102 CS42CJ 44446207 IC50 = 10230 nM T67102 C7VX1Q 44446209 IC50 = 5620 nM T67102 CG4N8T 44446210 IC50 = 5890 nM T67102 C1HZ9O 44446211 IC50 = 26300 nM T67102 CN2AB7 44446212 IC50 = 46770 nM T67102 CH6G1V 44447299 IC50 > 100000 nM T67102 C8T6YF 44449299 IC50 = 0.5 nM T67102 CW0LK4 44449760 Ki = 1071 nM T67102 C5LJY9 44449874 Ki = 142 nM T67102 CHU63Z 44449992 Ki = 310 nM T67102 C7GQY6 44450048 Ki = 810 nM T67102 CL1SO0 44450074 Ki = 2053 nM T67102 C0GOH4 44450139 Ki = 135 nM T67102 C0EPX3 44450198 Ki = 151 nM T67102 C2PJ1L 44450200 Ki = 300 nM T67102 CXS7Y3 44454508 IC50 = 7940 nM T67102 C2QI1J 44454509 IC50 = 30015 nM T67102 CML29V 44454541 IC50 = 25630 nM T67102 CBS73X 44454542 IC50 > 100000 nM T67102 CJ0NI6 44454543 IC50 = 10000 nM T67102 C0XMF7 44454839 IC50 = 4570 nM T67102 CTY3G5 44454842 IC50 = 9277 nM T67102 CIFD60 44454874 IC50 = 5413 nM T67102 CP08GW 44454875 IC50 = 3090 nM T67102 CU9GD7 44454913 IC50 = 6170 nM T67102 C6XY2B 44454914 IC50 = 47080 nM T67102 C7OGW4 44454944 IC50 = 12300 nM T67102 C10PVS 44454945 IC50 = 430 nM T67102 C1FM6T 44455733 IC50 = 54200 nM T67102 CAGM05 44478390 IC50 = 9600 nM T67102 C9P3XR 44478656 IC50 = 63400 nM T67102 CA4W3P 44478657 IC50 = 150100 nM T67102 CX24EA 44478658 IC50 = 47400 nM T67102 CJ7AL5 44478659 IC50 = 15400 nM T67102 CC3VB8 44478660 IC50 = 95300 nM T67102 CI2X9B 44517765 Ki > 5000 nM T67102 C8QT4P 44517766 Ki > 5000 nM T67102 C7AFS5 44527662 IC50 = 43 nM T67102 CM0A8K 44532986 IC50 = 360 nM T67102 CLH74F 44565900 IC50 > 100000 nM T67102 CMIP10 44565901 IC50 > 100000 nM T67102 C70BXJ 44565925 IC50 > 100000 nM T67102 CS6YO0 44566187 IC50 > 100000 nM T67102 CSF17Z 44566188 IC50 > 100000 nM T67102 CJP3U5 44566195 IC50 > 100000 nM T67102 CUFJ57 44566196 IC50 = 42 nM T67102 CTA78Q 44588631 Ki = 15 nM T67102 C5L4NQ 44588632 Ki = 24 nM T67102 C2E4RJ 44588633 Ki = 730 nM T67102 CQ18CM 44588634 Ki = 360 nM T67102 C4WXC8 44588635 Ki = 430 nM T67102 C3WC1U 44588636 Ki = 180 nM T67102 CG42IK 44588637 Ki > 5000 nM T67102 CQAT24 44588638 Ki = 1950 nM T67102 CF0N6C 44588639 Ki = 440 nM T67102 CA6I3V 44588640 Ki = 930 nM T67102 C8DB1H 44588641 Ki = 350 nM T67102 CA5SD6 44588642 Ki > 5000 nM T67102 C3JY7V 44588643 Ki > 5000 nM T67102 C9LZ3U 44588644 Ki > 5000 nM T67102 CKEZ47 44588645 Ki > 5000 nM T67102 CB1Q4T 44588646 Ki = 570 nM T67102 CFY78K 44588647 Ki = 1500 nM T67102 CLF0E5 44588648 Ki > 5000 nM T67102 C5W7KN 44588649 Ki > 5000 nM T67102 C0GR5A 44596194 Ki > 10000 nM T67102 C3OL5Q 44596195 Ki > 10000 nM T67102 C3E5AZ 44624107 IC50 = 1140 nM T67102 CUIY75 44624171 IC50 > 10000 nM T67102 CT46YX 44624237 IC50 = 3980 nM T67102 C8A2VT 44624238 IC50 = 1150 nM T67102 CT65UM 44624240 IC50 = 1510 nM T67102 C6N3JL 44624304 IC50 > 10000 nM T67102 C7AB0L 44625098 IC50 = 1050 nM T67102 C5WU0H 44625099 IC50 = 250 nM T67102 CL4BZ5 44625321 IC50 = 1230 nM T67102 C9ZGM1 44625323 IC50 = 250 nM T67102 CIO27W 44625397 IC50 = 230 nM T67102 CGX41M 44631838 Ki = 1100 nM T67102 CHL19P 44631842 IC50 = 1 nM T67102 CQ9G6O 44631933 IC50 = 820 nM T67102 C3M7ZG 45105274 Ki = 200 nM T67102 CJ0Y1O 45254127 IC50 = 640 nM T67102 CQB45G 45254505 IC50 = 1000 nM T67102 C1R3PL 45254506 IC50 = 3190 nM T67102 C2JD1Y 45254508 IC50 = 3390 nM T67102 C2YE7A 45254510 IC50 = 2300 nM T67102 CF92SD 45255915 IC50 = 9120 nM T67102 CA5YG0 45256104 IC50 = 29700 nM T67102 C0H9YA 45256107 IC50 = 37000 nM T67102 CRB2J3 45256108 IC50 = 13700 nM T67102 C43HDC 45256109 IC50 = 1100 nM T67102 C2Q3MJ 45256294 IC50 = 4470 nM T67102 C61DTC 45259043 IC50 = 9 nM T67102 C8BYZ2 45259044 IC50 = 240 nM T67102 CIY5X1 45267880 IC50 = 1570 nM T67102 CD2MC1 45268670 IC50 = 130 nM T67102 C16WVK 45269615 IC50 = 2900 nM T67102 C6JFK8 45277565 IC50 = 210 nM T67102 CVPF48 45277566 IC50 = 0.63 nM T67102 C6S2BO 45277567 IC50 > 5000 nM T67102 CJVC29 45277727 IC50 > 5000 nM T67102 CFY29M 45482524 Ki > 10000 nM T67102 CBC9V5 45482525 Ki > 10000 nM T67102 C7AF2S 45482526 Ki > 10000 nM T67102 CT0C5B 45482527 Ki > 10000 nM T67102 CX89VL 45482528 Ki > 10000 nM T67102 CXJU16 45482529 Ki > 10000 nM T67102 C14OFW 45482530 Ki > 10000 nM T67102 CF56XN 45482531 Ki > 10000 nM T67102 C1C6VB 45486934 IC50 = 2327 nM T67102 CF1RV5 45486939 IC50 > 10000 nM T67102 CTX69D 45486942 IC50 > 10000 nM T67102 CD0S3I 45486943 IC50 = 180 nM T67102 CEWV96 45486944 IC50 = 2300 nM T67102 C79FXL 45486945 IC50 = 2300 nM T67102 CUS3W8 45486946 IC50 = 9800 nM T67102 C04CSV 45486950 IC50 = 430 nM T67102 C3E5LA 45486952 IC50 = 450 nM T67102 CIM9P8 45486956 IC50 = 4300 nM T67102 CRO40Q 45486957 IC50 = 3900 nM T67102 CZU54V 45486959 IC50 = 330 nM T67102 C2O9HI 45486960 IC50 = 1400 nM T67102 CZDO08 45486961 IC50 = 80 nM T67102 CO24SK 45486962 IC50 = 84 nM T67102 CA2B9J 45486963 IC50 > 10000 nM T67102 C5YI3E 45486972 IC50 = 28 nM T67102 CG16NB 45486973 IC50 = 530 nM T67102 CB70SF 45486975 IC50 = 130 nM T67102 CO4NR2 45486979 IC50 = 22 nM T67102 CPYS43 45486980 IC50 = 670 nM T67102 C98DLY 45486981 IC50 = 3.3 nM T67102 C8E2PU 45486982 IC50 = 640 nM T67102 CROV56 45486983 IC50 = 2000 nM T67102 C8JQ7T 45486984 IC50 = 4400 nM T67102 C36ZXE 45486988 IC50 = 410 nM T67102 C1HK5L 45486991 IC50 = 170 nM T67102 CD9IL6 45486996 IC50 > 10000 nM T67102 CS5D9N 45486998 IC50 = 130 nM T67102 CS60MQ 45486999 IC50 = 4900 nM T67102 CKO57E 45487000 IC50 = 90 nM T67102 CB3D5J 45487001 IC50 = 3100 nM T67102 CF9IZ0 45487004 IC50 = 330 nM T67102 CR90BO 45487005 IC50 = 7200 nM T67102 C4NTM7 45488098 IC50 = 13370 nM T67102 CT95YJ 45488099 IC50 = 20780 nM T67102 C6W8LK 45488101 IC50 = 6220 nM T67102 CHMZ65 45488102 IC50 = 11100 nM T67102 CT51JC 45488104 IC50 = 9210 nM T67102 C1Q9DK 45488105 IC50 = 2710 nM T67102 CJ13RL 45488106 IC50 = 11570 nM T67102 CH7SG2 45488107 IC50 = 8550 nM T67102 CL0H9O 45488108 IC50 = 13140 nM T67102 CJ75VZ 45488110 IC50 = 26180 nM T67102 C4QV8Z 45488111 IC50 = 3150 nM T67102 C4ZD5W 45488112 IC50 = 2050 nM T67102 CXG2R1 45488113 IC50 = 69180 nM T67102 C8FTJ3 45488115 IC50 = 38180 nM T67102 CB10OE 45488116 IC50 = 4430 nM T67102 CE1ZX5 45488119 IC50 = 2600 nM T67102 CKBT31 45488120 IC50 = 4180 nM T67102 CH0W9R 45488121 IC50 = 2410 nM T67102 COT0P1 46178810 IC50 = 1176 nM T67102 CVW76R 46190732 IC50 = 3 nM T67102 CZ0JD1 46191766 IC50 = 11 nM T67102 C3VYC6 46217866 IC50 = 150 nM T67102 CH2EI5 46218828 Ki = 4300 nM T67102 CM9ON2 46225154 IC50 = 156 nM T67102 CK3O2Q 46231555 IC50 = 54000 nM T67102 CKE7B8 46233417 Ki = 840 nM T67102 C1EH4N 46233418 Ki = 1100 nM T67102 CD6EK4 46233419 Ki = 460 nM T67102 C8HX0R 46233420 Ki > 5000 nM T67102 CF5IV9 46233421 Ki > 5000 nM T67102 CPKS32 46233422 Ki > 5000 nM T67102 CD8IS3 46233423 Ki > 5000 nM T67102 CETW51 46233424 Ki > 5000 nM T67102 CU3EI0 46233611 Ki = 62 nM T67102 C0B6LM 46233613 Ki > 5000 nM T67102 C4IP1B 46233614 Ki > 5000 nM T67102 CHA57O 46233615 Ki > 5000 nM T67102 CG30XW 46233616 Ki > 5000 nM T67102 CA4IM2 46236672 IC50 = 50 nM T67102 C23TKX 46236812 IC50 = 50 nM T67102 CLX98O 46236813 IC50 = 50 nM T67102 CIZD19 46236814 IC50 = 50 nM T67102 CZK5E9 46238536 IC50 = 42000 nM T67102 C6KN1D 46830239 IC50 = 5500 nM T67102 CNP2S7 46844428 IC50 = 120 nM T67102 C7D4SK 46844429 IC50 = 410 nM T67102 CA3RK8 46881101 IC50 > 5000 nM T67102 CR8CP9 46881519 IC50 = 35 nM T67102 CC0V6G 46881567 IC50 = 48 nM T67102 CO5QC2 46881646 IC50 = 170 nM T67102 C7C2EK 46881691 IC50 = 7900 nM T67102 CWB9C6 46881692 IC50 = 7100 nM T67102 CJN4Y2 46881693 IC50 = 560 nM T67102 CS0O9T 46883935 IC50 = 13100 nM T67102 CDO30L 46883936 IC50 = 26400 nM T67102 C7O3XP 46884002 IC50 = 17400 nM T67102 C76UEW 46891887 IC50 = 395 nM T67102 CY36NG 46927945 IC50 = 140 nM T67102 CHT53N 49797544 IC50 = 3900 nM T67102 CD4W0Y 49797545 IC50 = 2340 nM T67102 CBW81T 49800161 IC50 = 14 nM T67102 CTP13K 49831178 IC50 = 490 nM T67102 CR41SW 49863021 IC50 = 1700 nM T67102 C9O7UP 49863022 IC50 = 6200 nM T67102 C9OWG2 49863023 IC50 = 2400 nM T67102 CNC25U 49863024 IC50 = 600 nM T67102 CED4S9 49863025 IC50 = 12000 nM T67102 CCY4G0 49863026 IC50 = 30000 nM T67102 C8T0LZ 49863027 IC50 = 3500 nM T67102 CSYU53 49863028 IC50 = 12000 nM T67102 C64OTC 49863029 IC50 = 6600 nM T67102 CWP2N9 49863030 IC50 = 2200 nM T67102 CWK1B5 49863031 IC50 = 1860 nM T67102 CVD2Q3 50898620 IC50 > 100000 nM T67102 C92SGN 50937466 IC50 = 6400 nM T67102 CD64NT 51039270 IC50 > 1000000 nM T67102 CJ6M8H 52940810 IC50 = 4200 nM T67102 C3DN8M 52940827 IC50 = 1170 nM T67102 CVT4K3 52940915 IC50 = 31560 nM T67102 CLM4T9 52941346 IC50 = 379 nM T67102 C5ZAD4 52941347 IC50 = 850 nM T67102 C5M2TI 52941360 IC50 = 411 nM T67102 CD4Y3W 52941431 IC50 = 42 nM T67102 CI4RQ0 52941475 IC50 = 9 nM T67102 CLJ01Q 52942108 IC50 = 300 nM T67102 CKU60L 52942135 IC50 = 480 nM T67102 CAOU31 52942213 IC50 = 480 nM T67102 C4G9QN 52942282 IC50 = 150 nM T67102 CX16LC 52942291 IC50 = 116710 nM T67102 CI8CX5 52942524 IC50 = 220 nM T67102 CEJ80Q 52942712 IC50 = 32 nM T67102 CVG51P 52942779 IC50 = 12170 nM T67102 CHN91J 52942848 IC50 = 4120 nM T67102 C4DWX6 52943931 IC50 = 263 nM T67102 C5QA0I 52943965 IC50 = 310 nM T67102 CFX8M2 52944038 IC50 = 67 nM T67102 C9MLZ6 52944049 IC50 = 29 nM T67102 C7J3ZR 52944055 IC50 > 10000 nM T67102 CQPD40 52944421 IC50 = 6200 nM T67102 C4PVH3 52944685 IC50 = 610 nM T67102 C8B2TR 52944893 IC50 = 8 nM T67102 C7W3MN 52945011 IC50 = 1050 nM T67102 CJL20O 52945191 IC50 = 140 nM T67102 C58HOG 52945584 IC50 = 3470 nM T67102 C0JQT1 52945785 IC50 = 380 nM T67102 CP4WO3 52945841 IC50 = 45 nM T67102 CQ4V8R 52946545 IC50 = 2600 nM T67102 C4QLW2 52946836 IC50 = 105 nM T67102 C6D8PN 52946837 IC50 = 1950 nM T67102 CO16KF 52946886 IC50 = 720 nM T67102 CIM9B8 52946887 IC50 = 3080 nM T67102 CRIQ87 52946950 IC50 = 3150 nM T67102 CWC0D6 52946966 IC50 = 2360 nM T67102 CK2TW7 52947058 IC50 = 1500 nM T67102 CG8AI7 52947059 IC50 = 200 nM T67102 CAL2H1 52947347 IC50 = 12 nM T67102 C5UV2T 52947441 IC50 = 4420 nM T67102 C43VCX 52947515 IC50 = 55 nM T67102 C45HZM 52948018 IC50 = 47 nM T67102 C6IC7P 52948105 IC50 = 12 nM T67102 CB3NQ0 52948140 IC50 = 1150 nM T67102 CY34UI 52948154 IC50 = 3500 nM T67102 CKT0J6 52948174 IC50 = 9900 nM T67102 CX4JT5 52948286 IC50 = 750 nM T67102 CHIL29 52948341 IC50 = 160 nM T67102 C9QI2S 52948682 IC50 = 24 nM T67102 C8YOD0 52948683 IC50 = 530 nM T67102 CQS24C 52948726 IC50 = 42 nM T67102 CPR34K 52948727 IC50 = 1720 nM T67102 C15VEP 52948732 IC50 = 40 nM T67102 CZ0DX7 52949259 IC50 > 200000 nM T67102 CIT74G 52949295 IC50 = 90 nM T67102 C12DGV 52949296 IC50 = 3110 nM T67102 CAGS10 52949452 IC50 = 1200 nM T67102 C2XIY3 52949466 IC50 = 2200 nM T67102 C5O9AP 52949507 IC50 = 500 nM T67102 CA56UD 52949889 IC50 = 125 nM T67102 CM7A0X 52949992 IC50 = 276 nM T67102 C25NMI 52949993 IC50 = 228 nM T67102 CPO5A7 52950127 IC50 = 4800 nM T67102 CKQ34B 52950166 IC50 = 245 nM T67102 C7IJ2F 53232612 IC50 > 10000 nM T67102 C70NYJ 53236891 IC50 = 510 nM T67102 C3DIM5 53316912 Ki = 460 nM T67102 CQA2R7 53318217 Ki = 0.75 nM T67102 CI4O5J 53320863 Ki = 13 nM T67102 C5AZH3 53322198 Ki = 200 nM T67102 CWUZ14 53322199 Ki = 1700 nM T67102 C9O2CI 53324843 Ki > 5000 nM T67102 C61FYW 53326116 Ki = 760 nM T67102 CXY4G5 53326117 Ki > 5000 nM T67102 CPRZ03 53464941 IC50 = 2220 nM T67102 C6K5JY 53464945 IC50 = 140 nM T67102 CH9CX8 53465067 IC50 = 1080 nM T67102 C17GML 53465141 IC50 = 93 nM T67102 CM62ZA 53465787 IC50 = 108000 nM T67102 C2RU1J 53493350 IC50 = 1894 nM T67102 C17NYM 53493353 IC50 = 1665 nM T67102 CZ7UV6 53493354 IC50 = 10144 nM T67102 C86VQT 53494150 IC50 = 59798 nM T67102 C2GUC3 53494692 IC50 = 1760 nM T67102 C1T6KF 53494828 IC50 = 3983 nM T67102 CF40KI 54580003 IC50 = 5890 nM T67102 CXF10V 54580145 IC50 = 2100 nM T67102 C3ROW7 54583129 IC50 = 7100 nM T67102 CB41FM 54583130 IC50 = 420 nM T67102 CO6T7C 54584085 IC50 = 900 nM T67102 C6C2NO 54585055 IC50 = 370 nM T67102 C7KU6J 54586032 IC50 = 4700 nM T67102 CY58NP 54586033 IC50 = 670 nM T67102 CAH7Y1 54681312 IC50 > 40000 nM T67102 C3P8YE 54681383 IC50 > 40000 nM T67102 CG1D6V 56658432 IC50 = 12980 nM T67102 C0RMT9 56658435 IC50 = 360 nM T67102 C2J7TS 56658436 IC50 = 26400 nM T67102 CW8IY4 56658437 IC50 = 31650 nM T67102 C45YJU 56658717 IC50 = 7400 nM T67102 CS4MX1 56658718 IC50 = 3800 nM T67102 CM4P2G 56661917 IC50 = 4790 nM T67102 C4QD7Z 56661918 IC50 = 29920 nM T67102 C47HVP 56661919 IC50 = 8000 nM T67102 CQP28A 56665390 IC50 = 1790 nM T67102 CXW4B7 56668819 IC50 = 1420 nM T67102 C1Z7MG 56668820 IC50 = 23800 nM T67102 C10MSR 56668821 IC50 = 2500 nM T67102 C5VIR4 56669107 IC50 = 28300 nM T67102 C1DFQ6 56672294 IC50 = 17300 nM T67102 CFE52J 56672296 IC50 = 13120 nM T67102 C2EZ8O 56672297 IC50 = 4850 nM T67102 CGNH26 56672298 IC50 = 13050 nM T67102 CCG59L 56672299 IC50 = 2200 nM T67102 CLP36K 56672300 IC50 = 18600 nM T67102 C43PXS 56675689 IC50 = 6690 nM T67102 CL8PK3 56675694 IC50 = 11800 nM T67102 CV3BE8 56675695 IC50 = 33000 nM T67102 CUI46G 56675696 IC50 = 4100 nM T67102 CO7G3P 56678998 IC50 = 830 nM T67102 C65LKQ 56678999 IC50 = 38650 nM T67102 CLW2C5 56679000 IC50 = 12800 nM T67102 CH80FW 56679262 IC50 = 54400 nM T67102 CGL67Z 56682312 IC50 = 4400 nM T67102 C07EXO 56682313 IC50 = 30500 nM T67102 CE8PW7 56682314 IC50 = 78400 nM T67102 C7QB6A 56682567 IC50 = 75800 nM T67102 C7SIV2 56834949 IC50 = 6212 nM T67102 CGZ0M9 56944167 IC50 > 300000 nM T67102 CH8FO4 56947420 IC50 = 6300 nM T67102 C4ZSQ1 56947421 IC50 = 840 nM T67102 CP2DE0 56947553 IC50 = 960 nM T67102 C6BW5Q 56947557 IC50 = 3200 nM T67102 C4K1XS 56947558 IC50 = 5400 nM T67102 C0NH9E 56947697 IC50 = 6200 nM T67102 CZ4M0T 56947699 IC50 = 1800 nM T67102 C7RZ0B 56947700 IC50 = 780 nM T67102 COHF14 56947701 IC50 = 11000 nM T67102 C0KY3J 56947828 IC50 = 940 nM T67102 C63PVB 56947829 IC50 = 600 nM T67102 CX3E4B 56948453 IC50 = 14000 nM T67102 CZ67RX 56948455 IC50 = 24000 nM T67102 C1TG8P 56948806 IC50 = 2300 nM T67102 C7K3BV 56950381 IC50 = 2000 nM T67102 C9Q4VL 57384270 IC50 = 1320 nM T67102 CDS03B 57384271 IC50 = 600 nM T67102 CBKI24 57384272 IC50 = 2530 nM T67102 C6IAW5 57384273 IC50 = 2810 nM T67102 C42JEK 57384274 IC50 = 510 nM T67102 C7DI1C 57385528 IC50 = 1390 nM T67102 CAR38J 57385530 IC50 > 10000 nM T67102 C90GLN 57385533 IC50 = 3750 nM T67102 CGPA23 57385772 IC50 = 1630 nM T67102 CU9FY0 57385773 IC50 = 5530 nM T67102 CA0X8R 57386049 IC50 = 1740 nM T67102 CLIW35 57386302 IC50 = 980 nM T67102 C5CF8I 57386304 IC50 = 290 nM T67102 CNAI80 57386563 IC50 = 2520 nM T67102 CB4WO2 57386811 IC50 = 340 nM T67102 C5VQE6 57386812 IC50 = 720 nM T67102 COL2R0 57386813 IC50 = 4160 nM T67102 CZT37N 57386814 IC50 = 7990 nM T67102 C0TOR5 57387067 IC50 = 1220 nM T67102 CG2R8K 57387068 IC50 = 1490 nM T67102 C1K6GV 57387069 IC50 = 2480 nM T67102 CI7LG6 57387070 IC50 = 1750 nM T67102 C52VTC 57387317 IC50 = 1720 nM T67102 CU3C7S 57387318 IC50 = 5200 nM T67102 C2HV9X 57387319 IC50 = 4370 nM T67102 C46BLJ 57387320 IC50 = 360 nM T67102 C67AEU 57387579 IC50 = 510 nM T67102 C7ZHD4 57387580 IC50 = 2000 nM T67102 CSC27H 57387581 IC50 = 2300 nM T67102 CD36BM 57387582 IC50 = 1030 nM T67102 CB5V0D 57387583 IC50 = 540 nM T67102 C5QXU9 57387806 IC50 = 2000 nM T67102 CFD9V5 57387807 IC50 = 690 nM T67102 C9DEX6 57387808 IC50 = 2400 nM T67102 CZ0W8T 57387809 IC50 = 450 nM T67102 CWLJ62 57387810 IC50 = 2220 nM T67102 C3MNK4 57388037 IC50 = 480 nM T67102 CYL8B2 57388039 IC50 > 10000 nM T67102 CP9V7X 57388040 IC50 = 3710 nM T67102 CJA0T7 57388041 IC50 = 3070 nM T67102 C0D8IE 57393022 IC50 = 21200 nM T67102 CO8JG5 57393023 IC50 = 44500 nM T67102 C28QVA 57398293 IC50 = 28500 nM T67102 CO2FV3 57398294 IC50 = 39200 nM T67102 CNV5E0 57398295 IC50 = 17800 nM T67102 C71GLZ 57401740 IC50 = 31900 nM T67102 C80LNE 57403473 IC50 = 21200 nM T67102 C1FTY8 57512157 IC50 = 126 nM T67102 C3G2ZX 57515809 IC50 = 465 nM T67102 CC8U3J 57825146 IC50 = 47700 nM T67102 CTU5I7 57825223 IC50 > 100000 nM T67102 CH94PW 57825229 IC50 > 100000 nM T67102 C0PID6 57843652 Ki = 53300 nM T67102 CWQ9B4 57844200 Ki > 100000 nM T67102 C6WU7P 57844259 Ki = 7100 nM T67102 CD9A1M 57844562 Ki = 63500 nM T67102 CU1FR6 58423762 IC50 = 97740 nM T67102 CC8TK0 58466119 IC50 = 660 nM T67102 C6QJX4 58466300 IC50 = 440 nM T67102 CJTL53 58909353 IC50 = 429 nM T67102 C3VHC7 59028115 IC50 = 8 nM T67102 CW63FG 59262280 Ki > 100000 nM T67102 CFD96H 59262349 Ki = 3500 nM T67102 CQO7U1 59262351 Ki = 2400 nM T67102 C1Y6QS 59262353 Ki = 6900 nM T67102 CC5J3G 59262483 Ki = 3800 nM T67102 C6Q4EZ 59262553 Ki = 8500 nM T67102 CID2C7 59262561 Ki = 2500 nM T67102 C2PJ4N 59271992 IC50 > 30000 nM T67102 CBH8L1 59388200 Ki = 6000 nM T67102 CP25LG 60043779 IC50 = 68 nM T67102 CQW7A8 60149247 Ki = 180 nM T67102 COXS42 60168050 IC50 = 577 nM T67102 CV43HQ 60168051 IC50 > 40000 nM T67102 C9E4NW 60202322 IC50 = 3 nM T67102 CUE46I 66575069 IC50 = 5.84 nM T67102 CCN98R 66649578 IC50 = 290 nM T67102 CHS2G5 66649612 IC50 = 9680 nM T67102 C75DVR 66649674 IC50 = 750 nM T67102 C2BGY7 66649788 IC50 = 3570 nM T67102 CFML30 66665322 IC50 > 250000 nM T67102 CB6ZA3 66683197 IC50 = 48603 nM T67102 C83LNT 66683198 IC50 = 11844 nM T67102 C8N2ZT 66683200 IC50 = 29540 nM T67102 CGKU53 66683659 IC50 = 88464 nM T67102 C92SYT 66683709 IC50 = 1259 nM T67102 CWE7G3 66683751 IC50 = 44161 nM T67102 CP09ND 66684067 IC50 = 624 nM T67102 C9AZ1X 66684136 IC50 = 5166 nM T67102 C7Z6OV 66684147 IC50 = 990 nM T67102 C7X6FL 66684245 IC50 = 8096 nM T67102 C1X4GA 66684386 IC50 = 9034 nM T67102 CGC47N 67236442 IC50 = 1717 nM T67102 C4V3NK 67246237 IC50 = 16800 nM T67102 CM8PJ4 67246553 IC50 = 26900 nM T67102 CYK23N 67246725 IC50 = 20100 nM T67102 CYA5T3 67246787 IC50 = 13700 nM T67102 C7R0IM 67247796 IC50 > 40000 nM T67102 CIT9Y0 67247849 IC50 = 30900 nM T67102 C63VKT 67247971 IC50 = 37300 nM T67102 CV2W4A 67248528 IC50 = 13800 nM T67102 C1DXK4 67248938 IC50 = 16000 nM T67102 COGX71 67249135 IC50 > 40000 nM T67102 CI1MQ0 67304745 IC50 = 8 nM T67102 C5X3ZN 67306893 IC50 = 4 nM T67102 CQ24FC 67950181 IC50 = 69000 nM T67102 CC69RG 67950202 IC50 = 140000 nM T67102 C2P8SB 67950244 IC50 = 7500 nM T67102 CBOC21 67970433 IC50 = 57000 nM T67102 C9TXI4 67970604 IC50 = 11000 nM T67102 C7KX8J 67970675 IC50 > 200000 nM T67102 CH9WP7 67970677 IC50 = 12000 nM T67102 C0IG9N 67970973 IC50 > 200000 nM T67102 C89UJX 67971074 IC50 > 200000 nM T67102 CSK05E 67971135 IC50 = 15000 nM T67102 C25BUR 67971352 IC50 = 3700 nM T67102 C8ZEP9 67971363 IC50 = 170000 nM T67102 C2SA9C 67971406 IC50 = 42000 nM T67102 CQ93MO 67971614 IC50 = 120000 nM T67102 C29ONK 67971826 IC50 = 47000 nM T67102 C8HEF1 67971920 IC50 = 76000 nM T67102 C7XBG9 68321727 IC50 = 2069 nM T67102 C5IP2Z 68321730 IC50 = 1030 nM T67102 CLZG95 68321802 IC50 = 627 nM T67102 CN3GX2 68321815 IC50 = 1085 nM T67102 C90AYO 68321837 IC50 = 265 nM T67102 CCKG03 68321840 IC50 = 683 nM T67102 CBY7W2 68321854 IC50 = 14704 nM T67102 CZM1N6 68321874 IC50 = 4368 nM T67102 CGZP43 68321882 IC50 = 300 nM T67102 CVH4Z8 68321895 IC50 = 6340 nM T67102 CT20FH 68321898 IC50 = 430 nM T67102 CR4W5M 68321900 IC50 = 3462 nM T67102 C9RS4D 68321905 IC50 = 447 nM T67102 C9B5LG 68321915 IC50 = 8611 nM T67102 C4LFD5 68321923 IC50 = 21 nM T67102 CGO28J 68321924 IC50 = 3709 nM T67102 C84FKJ 68321947 IC50 = 973 nM T67102 CFTJ53 68322072 IC50 = 249 nM T67102 C0TZ4R 68322076 IC50 = 735 nM T67102 CLNG90 68322078 IC50 = 798 nM T67102 CA15JL 68322079 IC50 = 2292 nM T67102 C81GAK 68322085 IC50 = 2513 nM T67102 CP98HL 68322184 IC50 = 6760 nM T67102 C7I8VG 68322203 IC50 = 420 nM T67102 CA1S5U 68432286 IC50 > 100000 nM T67102 C56CFA 68448803 IC50 > 10000 nM T67102 CX1W5L 68694228 IC50 > 40000 nM T67102 CQG75W 68696955 IC50 = 5 nM T67102 C53IHQ 68696989 IC50 = 36 nM T67102 CD0B4L 68697749 IC50 = 20500 nM T67102 C60VEF 68699589 IC50 = 46 nM T67102 CDQE76 70132509 Ki = 19453 nM T67102 CTO36I 70680446 IC50 = 50 nM T67102 CDX40V 70680447 IC50 = 11.3 nM T67102 C9F1QE 70680448 IC50 = 54.1 nM T67102 CCZ5J0 70681598 IC50 = 695 nM T67102 COE50A 70681599 IC50 = 347 nM T67102 CG4DK9 70682176 IC50 > 300000 nM T67102 C5W9EM 70682473 IC50 = 220 nM T67102 C1Y4QJ 70682474 IC50 = 300 nM T67102 CV84NM 70684257 IC50 > 300000 nM T67102 CATH92 70684290 IC50 > 300000 nM T67102 CJ4ZN8 70686411 IC50 > 300000 nM T67102 C9APE1 70686436 IC50 > 300000 nM T67102 CH35YM 70687977 IC50 = 2 nM T67102 CHD86L 70687986 IC50 = 12 nM T67102 CIA5Q8 70688505 IC50 > 300000 nM T67102 C8WBS4 70688511 IC50 > 300000 nM T67102 CMQ0T5 70690011 IC50 = 4 nM T67102 C3KTC7 70690563 IC50 > 300000 nM T67102 CQW43C 70690565 IC50 > 300000 nM T67102 C7CJ9K 70690592 IC50 > 300000 nM T67102 CDJ15O 70690877 IC50 = 540 nM T67102 CR57LJ 70692159 IC50 = 8 nM T67102 CFU45O 70694765 IC50 > 300000 nM T67102 CTUQ03 70696214 Ki = 27 nM T67102 CT25CI 70696325 IC50 = 11 nM T67102 C1H5VR 70696798 IC50 > 300000 nM T67102 C7O5IT 71268741 IC50 > 81000 nM T67102 CZ9LT5 71268850 IC50 > 100000 nM T67102 CEV0B7 71449561 Ki = 9.9 nM T67102 C21OKC 71449973 IC50 > 40000 nM T67102 CUIL24 71449974 IC50 > 40000 nM T67102 C86RHK 71451365 Ki > 5000 nM T67102 CIF8L6 71451795 IC50 = 7650 nM T67102 C49JDX 71451915 Ki = 7100 nM T67102 CDQ09Y 71452058 IC50 = 7.81 nM T67102 CN26XZ 71452059 IC50 = 3480 nM T67102 CA3H9D 71452060 IC50 = 7590 nM T67102 C2UC7A 71452061 IC50 = 20.9 nM T67102 CJ8IK3 71452990 IC50 = 700 nM T67102 C3X9OY 71453618 IC50 = 35700 nM T67102 CPOW01 71453619 IC50 > 40000 nM T67102 CEB6T9 71453620 IC50 = 3700 nM T67102 CTV35W 71453879 IC50 = 412 nM T67102 CLE7P2 71453880 IC50 = 0.0783 nM T67102 CO67FA 71453881 IC50 = 0.126 nM T67102 C4IOH6 71455340 IC50 = 28500 nM T67102 C8J1LO 71455341 IC50 = 44200 nM T67102 C2NM4Q 71455471 Ki = 8264 nM T67102 C93BQC 71455611 IC50 = 89.3 nM T67102 CWA79L 71457260 Ki = 690 nM T67102 CL2S3Y 71457261 Ki = 2000 nM T67102 CK73LU 71457396 IC50 = 17.3 nM T67102 CNM98L 71458534 Ki = 36 nM T67102 CM80QT 71458988 IC50 > 40000 nM T67102 CLG93R 71459108 Ki = 530 nM T67102 C3MV5B 71460183 IC50 = 4.5 nM T67102 CV0E9B 71460380 Ki = 120 nM T67102 CBO2M4 71460381 Ki = 750 nM T67102 C6OC0Z 71460382 Ki = 37 nM T67102 C1PRD6 71461037 IC50 = 71.7 nM T67102 C9L1IU 71461038 IC50 = 254 nM T67102 CP6IV2 71462074 Ki = 240 nM T67102 CD4QU0 71462075 Ki = 5000 nM T67102 C50VTC 71462510 IC50 > 40000 nM T67102 C0GBL7 71466345 IC50 > 100000 nM T67102 C5DTE9 71520763 IC50 = 1150 nM T67102 C3RS8D 71581444 IC50 = 370 nM T67102 CJ9S3O 71581445 IC50 = 72 nM T67102 C89CZA 71598542 IC50 = 890 nM T67102 C6N4LP 71598543 IC50 > 10000 nM T67102 CHK9Y2 71624098 IC50 = 185 nM T67102 CO3YI9 71624343 IC50 = 16820 nM T67102 CYQI35 71624345 IC50 = 37940 nM T67102 CIC4L2 71624469 IC50 = 49700 nM T67102 CA9Y2O 71624470 IC50 = 1606 nM T67102 CIU5Q1 71624579 IC50 = 2829 nM T67102 C7Z3GY 71624580 IC50 = 180420 nM T67102 C2MSD3 71624581 IC50 = 477 nM T67102 C4NHO5 71624685 IC50 = 603 nM T67102 CI6N2U 71624686 IC50 = 404 nM T67102 C5A6UZ 71624687 IC50 = 3072 nM T67102 CMN85D 71624688 IC50 = 1224 nM T67102 CI5P2V 71624689 IC50 = 329 nM T67102 C6K3CN 71625880 IC50 = 295 nM T67102 CCUI41 71664591 IC50 = 870 nM T67102 CKX64V 71664592 IC50 > 10000 nM T67102 C54DZH 71714118 IC50 > 300000 nM T67102 CPI2B3 71726571 IC50 = 6.3 nM T67102 C8J4WK 71726572 IC50 = 230 nM T67102 C08CYJ 71726699 IC50 = 4.3 nM T67102 C38LNQ 71726700 IC50 = 54 nM T67102 CPX7C6 71726820 IC50 = 2 nM T67102 CN2V1S 71738909 Ki = 2700 nM T67102 COVS02 71812189 IC50 = 9400 nM T67102 CLE0M5 71814501 IC50 = 80 nM T67102 CF9Q6G 71814502 IC50 = 144 nM T67102 C8GBJ2 71814503 IC50 = 70 nM T67102 C8OAN7 71814504 IC50 = 478 nM T67102 CVFW51 71814680 IC50 = 145 nM T67102 C53EOF 71814681 IC50 = 286 nM T67102 C1W4ND 71814682 IC50 = 255 nM T67102 CTG12Z 71814683 IC50 = 18 nM T67102 C5NXB9 71815029 IC50 = 16 nM T67102 CGBA97 71815030 IC50 = 8 nM T67102 C1GFK3 71815031 IC50 = 59 nM T67102 C4DNQ3 71815032 IC50 = 374 nM T67102 C9UV7C 72190738 IC50 = 1780 nM T67102 CZ60LS 72191037 IC50 = 1240 nM T67102 C14GNR 72191038 IC50 = 1200 nM T67102 C20HKS 72191344 IC50 = 4030 nM T67102 C0C5QH 72191659 IC50 = 3290 nM T67102 CYEI57 72191660 IC50 = 3390 nM T67102 C36QKA 72191661 IC50 = 7900 nM T67102 C1Y8VS 72191976 IC50 = 780 nM T67102 CO28LK 72191977 IC50 = 6830 nM T67102 C5ZGJ6 72191978 IC50 > 10000 nM T67102 CU80HY 72547065 IC50 = 74900 nM T67102 CE3X8Y 72547066 IC50 = 13900 nM T67102 CCVG84 72547070 IC50 = 15700 nM T67102 CX70JT 72547320 IC50 = 13100 nM T67102 C5DC0Z 72946535 IC50 > 10000 nM T67102 C8K6NI 72946537 IC50 > 10000 nM T67102 CQM8U4 72946738 IC50 > 10000 nM T67102 CQ3DV8 72946943 IC50 > 10000 nM T67102 CYXC78 72947373 IC50 > 10000 nM T67102 CX34PN 73017594 IC50 = 2030 nM T67102 C43EOP 73345995 IC50 = 0.84 nM T67102 CEHO98 73345996 IC50 = 78 nM T67102 CMHA87 73346002 IC50 = 8.1 nM T67102 C1IFV6 73346019 IC50 = 362 nM T67102 C62BWK 73347547 IC50 = 1 nM T67102 CK40LM 73349243 IC50 = 2450 nM T67102 CR2JN8 73350632 IC50 = 29 nM T67102 C3ABQ1 73350653 IC50 = 2844 nM T67102 CSWI58 73350654 IC50 = 2 nM T67102 C2PLM7 73350655 IC50 = 77 nM T67102 CSM21F 73352126 IC50 < 2 nM T67102 CF0ST3 73355087 IC50 = 29 nM T67102 C74BWF 73355106 IC50 = 5 nM T67102 CVW0J5 73355107 IC50 = 6 nM T67102 C86UGE 73356659 IC50 < 2 nM T67102 C6VCF3 73356671 IC50 = 22506 nM T67102 C3BF0T 73356672 IC50 = 251 nM T67102 CX7P2O 73356673 IC50 = 74 nM T67102 CZ6Q1I 73388368 IC50 = 25100 nM T67102 CB7J0I 73507165 IC50 = 83100 nM T67102 CEP9F4 73507167 IC50 > 72000 nM T67102 C7Y5QC 73507384 IC50 > 91400 nM T67102 C97WEM 75593288 IC50 = 32000 nM T67102 CD4IX1 75593344 IC50 = 45000 nM T67102 CT8R2Z 76311036 IC50 = 490 nM T67102 CTG78Z 76311037 IC50 = 57000 nM T67102 C16WUE 76314667 IC50 = 810 nM T67102 C51UAX 76318242 IC50 = 4600 nM T67102 C4MF7L 76321932 IC50 = 1700 nM T67102 C31GTN 76329120 IC50 = 2600 nM T67102 COFK24 76332783 IC50 = 96000 nM T67102 CTJG92 76336403 IC50 = 160000 nM T67102 C3N9SR 76871907 IC50 = 1900 nM T67102 CTVA19 76871908 IC50 = 58 nM T67102 CQT14W 76955651 IC50 = 8000 nM T67102 C1BY0I 85470144 IC50 = 22000 nM T67102 CSM4C1 86288475 IC50 = 42 nM T67102 CV51KR 86288476 IC50 = 54 nM T67102 CB5F1W 86343364 IC50 = 140 nM T67102 CKG7N2 86343365 IC50 = 6600 nM T67102 C9IVM5 86343366 IC50 = 19300 nM T67102 CZ7Y0L 86658490 IC50 = 130000 nM T67102 C7OIC6 86762648 IC50 > 100000 nM T67102 CQCJ02 89512686 IC50 = 3870 nM T67102 CE7PH6 89997520 IC50 = 710 nM T67102 C2SJY8 89997744 IC50 = 1040 nM T67102 CFYO09 89997799 IC50 = 530 nM T67102 CT38QK 89998122 IC50 = 650 nM T67102 C7NA0W 89998237 IC50 = 4100 nM T67102 CVCR46 90285136 IC50 = 170 nM T67102 C0RM9Z 90285319 IC50 = 92 nM T67102 CD76NR 90285590 IC50 = 81 nM T67102 CD79MA 90285610 IC50 = 8.6 nM T67102 C9D5JT 90285792 IC50 = 44 nM T67102 CRNS50 90285861 IC50 = 690 nM T67102 CA7P0E 90285921 IC50 = 8300 nM T67102 C2ANE7 90285955 IC50 = 320 nM T67102 C9S7ZM 90285987 IC50 = 120 nM T67102 CIG87W 90286001 IC50 = 140 nM T67102 C79LYP 90294431 IC50 = 24 nM T67102 C75FIA 90294442 IC50 = 240 nM T67102 CP6WC9 90294647 IC50 = 370 nM T67102 C7PO1W 90308598 IC50 > 100000 nM T67102 C7OLJ6 90414780 IC50 = 1835 nM T67102 CS7ZM6 90655842 IC50 = 170 nM T67102 CQK42C 90655843 IC50 = 68 nM T67102 C64ASN 90655844 IC50 = 100 nM T67102 C65BUL 90655845 IC50 = 200 nM T67102 COG5V7 90655846 IC50 = 110 nM T67102 CL81MW 90655847 IC50 = 38 nM T67102 CAC0H4 90655848 IC50 = 500 nM T67102 CYS25V 90655849 IC50 = 19 nM T67102 CH9VJ1 90655850 IC50 = 32 nM T67102 CYV70Z 90655851 IC50 = 4400 nM T67102 CPGK89 90655852 IC50 = 120 nM T67102 C48HVL 90655853 IC50 = 5800 nM T67102 C4FR5P 90655854 IC50 = 40 nM T67102 C2GR6X 90655855 IC50 = 51 nM T67102 CL07NM 90655856 IC50 = 350 nM T67102 CXAP16 90655857 IC50 = 140 nM T67102 CAQ05V 90693645 Ki = 1.25 nM T67102 CUI10E 91666686 IC50 = 19100 nM T67102 C72FWD 91929322 Ki > 10000 nM T67102 CWZX73 91971958 IC50 >= 100000 nM T67102 C02GTW 102160610 IC50 = 87000 nM T67102 CZK0L7 105539825 IC50 = 4600 nM T67102 C1UXK6 117844010 IC50 = 1740000 nM T67102 C94WRZ 118435363 IC50 > 300000 nM T67102 C1WL4E 118435382 IC50 > 300000 nM T67102 C5L9VH 118435403 IC50 = 197600 nM T67102 CNXH97 118435407 IC50 > 97000 nM T67102 C8Z2FP 118435412 IC50 > 43000 nM T67102 CJIP45 118435414 IC50 = 163600 nM T67102 CY6EP7 118435506 IC50 > 96700 nM T67102 CPE35X 118435524 IC50 > 70300 nM T67102 CVK6Y8 118435560 IC50 > 300000 nM T67102 CN5L8K 118435601 IC50 > 95000 nM T67102 C37SFM 118435617 IC50 = 34800 nM T67102 CL6IV1 118440826 IC50 > 100000 nM T67102 CHIL17 118441142 IC50 > 100000 nM T67102 CSNR31 118576102 IC50 = 170 nM T67102 CM4TS0 118576345 IC50 = 98 nM T67102 C40ZTY 118583234 IC50 = 67 nM T67102 C81IOF 118586503 IC50 = 510 nM T67102 CQ5NK9 118709822 IC50 = 440 nM T67102 C4VDW0 118709823 IC50 = 1500 nM T67102 CDK81L 118709824 IC50 = 2700 nM T67102 CQM10N 118709825 IC50 = 3000 nM T67102 CXQD06 118709826 IC50 = 6100 nM T67102 CMZO04 118709827 IC50 = 10000 nM T67102 C86DZI 118709828 IC50 = 18000 nM T67102 C5MES8 118709829 IC50 = 25000 nM T67102 CAWM98 118709830 IC50 = 29000 nM T67102 CS39CI 118709831 IC50 = 280 nM T67102 CY9G8O 118716198 IC50 > 100000 nM T67102 CVJF59 118716317 Ki = 0.011 nM T67102 CA79YF 118716318 Ki = 0.0042 nM T67102 C3Q5BM 118716319 Ki = 0.00143 nM T67102 CI6H0V 118716320 Ki = 31 nM T67102 CL6TE3 118716321 IC50 > 100000 nM T67102 C4IZ7G 118716325 IC50 > 100000 nM T67102 CQB1N2 118716328 IC50 > 100000 nM T67102 CEU78H 118717559 IC50 > 100000 nM T67102 CCT87K 118717561 IC50 > 100000 nM T67102 CYR34C 118717562 IC50 > 100000 nM T67102 C3U5OB 118717564 IC50 > 100000 nM T67102 CSWB75 118717566 IC50 > 100000 nM T67102 C4FWD7 118717568 IC50 > 100000 nM T67102 CH87TO 118717570 IC50 > 100000 nM T67102 CXAF54 118717573 IC50 = 43 nM T67102 CVKR02 118717582 IC50 = 713 nM T67102 C5SZC4 118717584 IC50 = 447 nM T67102 C50AUM 118717586 IC50 = 5100 nM T67102 CHNF21 118717648 IC50 = 4800 nM T67102 C98MHD 118717651 IC50 > 100000 nM T67102 C1UGM6 118717653 IC50 = 29000 nM T67102 CMV83O 118717655 IC50 > 100000 nM T67102 CS0T9I 118717657 IC50 > 100000 nM T67102 C1BX8S 118717659 IC50 > 100000 nM T67102 C64WVI 118717661 IC50 > 100000 nM T67102 CIJ23K 118718355 Ki = 3500 nM T67102 C0EQ3L 118718356 Ki = 35 nM T67102 C4WHC8 118719663 Ki = 33000 nM T67102 C08UOL 118719664 Ki > 100000 nM T67102 CPT24G 118719665 Ki > 100000 nM T67102 CJW94R 118719666 Ki > 100000 nM T67102 CQ35DS 118719667 Ki > 100000 nM T67102 CP1R2J 118719668 Ki = 2800 nM T67102 CO2GZ4 118719669 Ki = 25500 nM T67102 CK1IT5 118719670 Ki = 44000 nM T67102 C5K9GN 118720051 Ki = 28000 nM T67102 CXUT34 118720052 Ki = 870 nM T67102 CRU2Q0 118720053 Ki = 8500 nM T67102 C50SLJ 118720054 Ki = 23000 nM T67102 C16QPS 118720056 Ki = 6000 nM T67102 C0YJ7W 118720058 Ki = 25000 nM T67102 CO1GD9 118720059 Ki = 7500 nM T67102 C3A6VB 118725861 IC50 = 5800 nM T67102 C3MNQ4 118725862 IC50 = 11600 nM T67102 C1TS2W 118725863 IC50 = 600 nM T67102 C1LTN0 118725864 IC50 = 680 nM T67102 C9EP7A 118732788 IC50 > 100000 nM T67102 CQD8B7 118732789 IC50 > 100000 nM T67102 C4HLF7 118732790 IC50 > 100000 nM T67102 C39IRT 118732791 IC50 = 63000 nM T67102 C4MTK9 118797904 IC50 = 99 nM T67102 C61QPW 118797905 IC50 = 1900 nM T67102 C5NE9P 118866030 IC50 = 1245000 nM T67102 COR8Y4 118866094 IC50 >= 750000 nM T67102 CELZ36 118866105 IC50 = 137000 nM T67102 CK2U6X 118866347 IC50 = 796000 nM T67102 C4MLU1 118866454 IC50 = 425000 nM T67102 CH6AT4 118866474 IC50 = 856000 nM T67102 CM2N6G 118866838 IC50 = 319000 nM T67102 CIM4Y6 118866963 IC50 = 400000 nM T67102 C9M2WU 118866986 IC50 = 48000 nM T67102 CT4Z2R 118884907 IC50 = 281000 nM T67102 CO7E4P 122180108 IC50 > 100000 nM T67102 CJM51V 122180111 IC50 = 277000 nM T67102 C15DUY 122180113 IC50 > 100000 nM T67102 C13ELK 122180115 IC50 > 300000 nM T67102 CXMQ41 122180117 IC50 = 797000 nM T67102 C2R6SY 122197438 IC50 = 26300 nM T67102 CDG6R0 122197443 IC50 = 2240 nM T67102 CK7W8B 123132907 IC50 = 32400 nM T67102 CRW0C2 123132915 IC50 > 100000 nM T67102 C45OVL 126693206 IC50 > 100000 nM T67102 C9QKI3 127020966 IC50 > 100000 nM T67102 C2XHZ8 127026505 IC50 = 53400 nM T67102 CB3X2O 127026506 IC50 = 9000 nM T67102 C3DIN6 127027428 IC50 = 25000 nM T67102 CJM2K9 127027429 IC50 = 19500 nM T67102 C9RKY8 127027430 IC50 = 9000 nM T67102 C5XU8O 127027434 IC50 = 2200 nM T67102 C51ONW 127027435 IC50 = 5000 nM T67102 CZ0M8K 127027436 IC50 = 3000 nM T67102 CR36NE 127027761 IC50 = 1400 nM T67102 CHBD07 127027762 IC50 = 8600 nM T67102 C7ZI6Q 127028384 IC50 = 100000 nM T67102 C7W8FM 127028385 IC50 = 3200 nM T67102 C2E3QR 127028386 IC50 > 100000 nM T67102 C9H3QY 127028711 IC50 = 220000 nM T67102 C5CR4Z 127028712 IC50 = 6000 nM T67102 CLGB70 127038526 IC50 > 200000 nM T67102 CAT8G7 127039677 IC50 = 91000 nM T67102 C9LAO0 127040014 IC50 = 52000 nM T67102 CCV17U 127044735 IC50 = 820 nM T67102 C9OTI7 127044896 IC50 = 470000 nM T67102 C7S2LA 127044941 IC50 = 197 nM T67102 CS3Z7A 127045094 IC50 = 58 nM T67102 CBU0D5 127050883 IC50 = 57 nM T67102 CZ48VN 132505928 IC50 = 380 nM T67102 CHE5R1 132505929 IC50 > 10000 nM T67102 C9W6JQ 135125856 IC50 = 35800 nM T67102 CKVF19 135126469 IC50 = 35800 nM T67102 CI1D7K 135875806 IC50 > 100000 nM T67102 CK3R8X 136219251 IC50 > 30000 nM T67102 C60STM 136219252 IC50 > 30000 nM T67102 C8L5PZ 137348437 IC50 = 480000 nM T67102 CLE04H 137348743 IC50 = 5900 nM T67102 C8JWF7 137633017 IC50 > 100000 nM T67102 CU40QT 137634377 IC50 = 65500 nM T67102 CLK7A3 137635011 IC50 > 100000 nM T67102 CY5M8Z 137635828 IC50 > 100000 nM T67102 C2B1MZ 137637375 IC50 > 100000 nM T67102 CEVA49 137637780 IC50 > 100000 nM T67102 CSQL63 137640486 IC50 > 100000 nM T67102 C91GMY 137641491 IC50 > 100000 nM T67102 C9BF0V 137643369 IC50 > 100000 nM T67102 CV56QL 137645221 IC50 > 100000 nM T67102 CG3U5K 137645264 Ki = 1500 nM T67102 CTB27V 137646126 IC50 > 100000 nM T67102 C10CBD 137646316 IC50 > 100000 nM T67102 CJXK40 137648425 IC50 > 100000 nM T67102 CVR29E 137651451 IC50 = 71800 nM T67102 C8HSX7 137652983 IC50 > 100000 nM T67102 CQ32NO 137653545 IC50 > 100000 nM T67102 CXY7F1 137654633 IC50 > 100000 nM T67102 CTU5C1 137656577 IC50 = 95300 nM T67102 C3L8WX 137657646 IC50 > 100000 nM T67102 C3YFL4 137662127 IC50 > 100000 nM T67102 C0JQU4 139589854 IC50 = 100 nM T67102 CF05LW 139589856 IC50 = 5.5 nM T67102 C31YCQ 139590075 IC50 = 270 nM T67102 C5XYE9 145864193 IC50 = 0.6 nM T67102 C8X5CM 145864195 IC50 = 5.8 nM T67102 C63WRI 145946134 IC50 = 2.5 nM T67102 C6HOU5 145950897 IC50 = 900 nM T67102 CU1VE4 145951062 IC50 = 1600 nM T67102 C4YMX8 145955472 IC50 = 50 nM T67102 CRA7P1 145958864 IC50 = 57 nM T67102 CJP34X 145965420 IC50 > 100000 nM T67102 C36CZY 145966369 IC50 > 100000 nM T67102 C0H5UD 145967429 IC50 > 100000 nM T67102 CSC48Q 145968177 IC50 = 13000 nM T67102 C24PUM 145968574 IC50 = 25000 nM T67102 CJ2V6B 145968904 IC50 = 93000 nM T67102 C8DOU5 145968976 IC50 = 11000 nM T67102 C1D6MG 145969118 IC50 = 3200 nM T67102 CT1V0I 145969327 IC50 = 71000 nM T67102 CYH45E 145970255 IC50 > 100000 nM T67102 CVAW24 145970337 IC50 = 430 nM T67102 CT57RL 145970338 IC50 = 400 nM T67102 CDR2G9 145970368 IC50 = 2700 nM T67102 CM8X7O 145970397 IC50 = 20000 nM T67102 CP8A0Z 145970407 IC50 = 29000 nM T67102 C4F6NT 145970582 IC50 > 100000 nM T67102 CH9P3X 145970804 IC50 = 100000 nM T67102 CZ3X4R 145970818 IC50 > 100000 nM T67102 CS64YI 145970835 IC50 = 21000 nM T67102 C53OSI 145971666 IC50 > 97000 nM T67102 CVK1O7 145974594 IC50 > 100000 nM T67102 CVM02B 145974600 IC50 > 64000 nM T67102 CKU21C 145977020 IC50 > 100000 nM T67102 CM27YI 145977049 IC50 > 98000 nM T67102 CYH46T 145978250 IC50 > 100000 nM T67102 CVK9J5 145978628 IC50 > 100000 nM T67102 CI4C2V 145980078 IC50 = 12000 nM T67102 CV6N5E 145980299 IC50 = 310000 nM T67102 CL2O0B 145980889 IC50 = 3600 nM T67102 C3BS5J 145981023 IC50 = 72000 nM T67102 C4XG5A 145983198 IC50 = 2700 nM T67102 C17GWT 145983210 IC50 = 15000 nM T67102 CWP2Q5 145986616 IC50 = 640000 nM T67102 CK9L8J 145987341 IC50 = 4400 nM T67102 C95VSG 145987742 IC50 > 100000 nM T67102 CNC1H3 145988728 IC50 = 1100000 nM T67102 C5PA1C 145988827 IC50 = 98000 nM T67102 CUGP43 145990468 IC50 = 4500 nM T67102 CZK41W 145990916 IC50 = 1200000 nM T67102 CN7I8T 145991278 IC50 = 660 nM T67102 CSAI70 145991785 IC50 = 1000000 nM T67102 CKVO52 155513754 IC50 = 1420 nM T67102 CE9RV3 155515912 IC50 = 100 nM T67102 C93IED 155516320 IC50 = 190 nM T67102 CM8U5I 155516895 IC50 = 3.1 nM T67102 CH72PJ 155517364 IC50 = 5200 nM T67102 COG03P 155518682 IC50 = 210 nM T67102 CAD6V5 155518995 IC50 = 120 nM T67102 C2S4ZM 155519404 IC50 = 7000 nM T67102 CW89FM 155520640 IC50 = 1000 nM T67102 C85GWP 155521302 IC50 = 700 nM T67102 CAD85F 155522348 IC50 = 600 nM T67102 C9ZVR0 155522599 IC50 = 1460 nM T67102 CA4N8E 155522934 IC50 = 32 nM T67102 C36PVM 155523018 IC50 = 11 nM T67102 C01LEB 155523479 IC50 = 270 nM T67102 CPEK52 155523929 IC50 = 1300 nM T67102 COG6S8 155524310 IC50 = 580 nM T67102 CJ1VB7 155524560 IC50 = 39 nM T67102 CTHW85 155525119 IC50 = 16 nM T67102 CG52WB 155525722 IC50 = 2500 nM T67102 C8BUC1 155525857 IC50 = 2000 nM T67102 CTKF74 155530540 IC50 = 3800 nM T67102 CLK7B5 155531254 IC50 = 68 nM T67102 CQV8H4 155533154 IC50 = 40 nM T67102 CWR61T 155534320 IC50 = 220 nM T67102 CW2N6T 155536787 IC50 = 15 nM T67102 CRN6V8 155537831 IC50 = 250 nM T67102 CUK21B 155538074 IC50 = 795000 nM T67102 C03KZX 155539456 IC50 = 400 nM T67102 CVBR73 155539645 IC50 = 2100 nM T67102 C16ZMF 155540206 IC50 = 150 nM T67102 CHQD90 155541280 IC50 = 18300 nM T67102 C25CXT 155542250 IC50 = 4900 nM T67102 CLW25Z 155542966 IC50 = 560 nM T67102 CM30ZB 155543610 IC50 = 340 nM T67102 CD6QL8 155545276 IC50 = 310 nM T67102 CK82SO 155547210 IC50 = 1660 nM T67102 C5FVL6 155547688 IC50 = 3.8 nM T67102 C51TEL 155548749 IC50 = 150 nM T67102 C5AMG2 155548757 IC50 = 55 nM T67102 C8GHP7 155550764 IC50 = 4.2 nM T67102 CGC20T 155551403 IC50 = 4800 nM T67102 CO9C7X 155552427 IC50 = 750 nM T67102 CI35JQ 155552899 IC50 = 96 nM T67102 CH95SX 155555744 IC50 = 27 nM T67102 CXK6V2 155555899 IC50 = 4.7 nM T67102 C2B8TR 155556406 IC50 = 262000 nM T67102 CMN6E1 155556535 IC50 = 760 nM T67102 C7DH9B 155556912 IC50 = 1997 nM T67102 CMR8O0 155557206 IC50 = 850 nM T67102 CF0R4Y 155557732 IC50 = 1.1 nM T67102 CJ7L5D 155558184 IC50 = 3.5 nM T67102 CUT69N 155558703 IC50 = 21 nM T67102 CGS42K 155558817 IC50 = 500 nM T67102 C9ZO7H 155558879 IC50 = 8.2 nM T67102 CW5TS8 155558999 IC50 > 200000 nM T67102 CCNM34 155560652 IC50 = 2250 nM T67102 C86SOP 155561681 IC50 = 15000 nM T67102 C5E9XF 155561692 IC50 = 500 nM T67102 C3XWV6 155562002 IC50 = 9 nM T67102 CT5C3X 155563480 IC50 = 22 nM T67102 C7E5VH 155565512 IC50 = 500 nM T67102 CYPV36 155565800 IC50 = 4400 nM T67102 CL6J1D 155566247 IC50 = 20 nM T67102 C1T2PI 155566542 IC50 = 67 nM T67102 CU42CE 155567829 IC50 > 100000 nM T67102 CBK7Z5 155568332 IC50 = 40 nM T67102 C45OJY 155568626 IC50 = 560 nM T67102 C3C1XH 11497497 IC50 = 910 nM T67102 CBQP67 11613166 IC50 = 300 nM T67102 C1KYA7 46877606 IC50 = 210 nM T67102 D00QMZ 44314223 Ki = 2400 nM T67102 D02LCH 16659106 Ki = 41 nM T67102 D07LUJ 64945 IC50 = 18200 nM T67102 D07NFJ 44314383 IC50 = 1200 nM T67102 D08AES 11578664 Ki = 3000 nM T67102 D08SCG 44327926 Ki = 1300 nM T67102 D08XLM 44314315 Ki = 1600 nM T67102 D09PZT 44297826 Ki = 210 nM T67102 D09SOY 15054176 IC50 > 100000 nM T67102 D0H3EJ 11205295 IC50 < 10 nM T67102 D0JI2X 44314268 Ki = 2100 nM T67102 D0KK6A 15126552 Ki = 3.2 nM T67102 D0P6RT 10078814 Ki = 18 nM T67102 D0S3BO 9895503 Ki = 2 nM T67102 D0S4BV 657149 IC50 = 20362 nM T67102 D0Y5IQ 44255320 IC50 = 40 nM T36935 CAEO59 752376 Ki = 300 nM T36935 CDXG58 9915884 IC50 = 226 nM T36935 CW5V7Y 44559839 IC50 = 13000 nM T36935 C1WF8N 45481867 Ki = 48.4 nM T36935 CP8IO2 45481868 Ki = 27.5 nM T36935 CCB46H 45481881 Ki = 25.3 nM T36935 C8L2QP 45481882 Ki = 2.5 nM T36935 C9S2LZ 45481883 Ki = 19.9 nM T36935 CF2AX3 45481884 Ki = 0.2 nM T36935 C8EKC7 45481885 Ki = 5.6 nM T36935 C9OCW6 45481886 Ki > 50 nM T36935 C5WUQ7 45481896 Ki = 65 nM T36935 CIPS79 45481897 Ki = 3.6 nM T36935 C5NEO7 45481898 Ki = 4.4 nM T36935 CL2XE8 45481899 Ki = 6.5 nM T36935 CUE83D 45481902 Ki = 11.9 nM T36935 CN3IR2 45481903 Ki = 12.8 nM T36935 C7ZW6S 45481904 Ki = 13.1 nM T36935 CT0QK2 45481905 Ki = 13.7 nM T36935 C0CQ5I 45481906 Ki = 18.6 nM T36935 C1EFL0 45481907 Ki = 21.8 nM T36935 CE8TK4 45481908 Ki = 29.4 nM T36935 CJ7PE0 45481909 Ki = 37.4 nM T36935 C7XC2E 45481910 Ki = 41.9 nM T36935 C06LNX 45481911 Ki > 50 nM T36935 CHDC31 45481912 Ki > 50 nM T36935 CVD7H2 45481913 Ki > 50 nM T36935 CF29EV 45481914 Ki > 50 nM T36935 C1G6JV 45481915 Ki > 50 nM T36935 CA4S1Q 45481916 Ki > 50 nM T36935 C3C9AY 45481917 Ki > 100 nM T36935 C1PGU4 45481918 Ki > 100 nM T36935 CUPK21 45481919 Ki > 100 nM T36935 CC5ED7 45481920 Ki > 500 nM T36935 C8H0FC 45481921 Ki > 500 nM T36935 CH25WT 45481923 Ki > 1000 nM T36935 CX8P3W 45481924 Ki > 1000 nM T36935 CT1IF2 45481925 Ki > 1000 nM T36935 CJD03W 45481926 Ki = 3.9 nM T36935 C0QY1E 45481927 Ki = 7.5 nM T36935 CBT01H 45481928 Ki = 8.8 nM T36935 C9N2ZV 45481929 Ki = 13.1 nM T36935 C6YCA1 45481930 Ki = 18.2 nM T36935 C5EMY7 45481931 Ki = 19.9 nM T36935 CCDX29 45481932 Ki = 25.9 nM T36935 C6A5WQ 45481933 Ki = 43.8 nM T36935 CI08ZL 45481934 Ki > 500 nM T36935 CG2S1H 45481935 Ki > 1000 nM T36935 CHT38O 45481936 Ki > 1000 nM T36935 CP68VG 45481937 Ki > 1000 nM T36935 CM8WF7 45481938 Ki > 1000 nM T36935 CR8AO5 70683138 IC50 = 226 nM T36935 CRMU86 71451729 Ki = 500 nM T36935 C4RZ8T 71680692 Ki = 164.5 nM T36935 CVF1P5 71680693 Ki = 24.23 nM T36935 CG9N3E 71680694 Ki = 43.05 nM T36935 C5F1YH 71680695 Ki = 22.01 nM T36935 C9RGE0 71680852 Ki = 302.1 nM T36935 C6B8UX 71680853 Ki = 310.29 nM T36935 CQB7X6 71680854 Ki = 52.11 nM T36935 C15EQX 71680855 Ki = 61.48 nM T36935 CUNX13 71681017 Ki = 73.33 nM T36935 CW2IL3 71681018 Ki = 64.41 nM T36935 COTQ71 71681171 Ki = 228.78 nM T36935 CC2QE7 71681172 Ki = 102.46 nM T36935 C50ATU 73345680 Ki > 500 nM T36935 CUT98E 73354917 Ki = 45000 nM T36935 D04BPQ 71681016 Ki = 72 nM T53389 D05ROI 44462760 IC50 = 3700 nM T53389 D06TFI 10090485 IC50 = 51 nM T53389 D0E3TC 44259 IC50 = 6870 nM T53389 D0MR0B 54766013 Ki = 6.296 nM T53389 D0F8DL 176155 IC50 = 6000 nM T53389 C9VW8M 449054 IC50 = 20 nM T53389 CO0AG7 453216 IC50 > 50000 nM T53389 CU0TP2 3539049 IC50 = 382 nM T53389 C9SB1M 4464598 IC50 = 355 nM T53389 C79ZDX 5287525 IC50 = 1320 nM T53389 CS5FX9 9836405 IC50 = 28 nM T53389 CQR6U0 9838979 IC50 = 47 nM T53389 CJ0GI8 9848057 IC50 = 25 nM T53389 C9L2KP 9858084 IC50 = 48 nM T53389 CY6LX3 9861063 IC50 = 107 nM T53389 CS5ZJ4 9863630 IC50 = 1500 nM T53389 CJF9D2 9880709 IC50 = 49 nM T53389 C63ZVC 9901964 IC50 = 24 nM T53389 C76AHX 9907180 IC50 = 2950 nM T53389 CLV0X4 9908131 IC50 = 170 nM T53389 CV61YK 9922527 IC50 = 40 nM T53389 C2S9NJ 9923039 IC50 = 6 nM T53389 CVZR49 9924137 IC50 > 20000 nM T53389 C9CRT7 9925372 IC50 = 24 nM T53389 C8V1ZH 9925495 IC50 = 10 nM T53389 CFS8T0 9944477 IC50 = 2620 nM T53389 CPH63X 9945516 IC50 = 43 nM T53389 CVA8M7 9946092 IC50 = 928 nM T53389 CWR08E 9947683 IC50 > 20000 nM T53389 C5HPV6 9951300 IC50 = 260 nM T53389 CFH9D2 9968513 IC50 = 1300 nM T53389 CY05UE 9969336 IC50 = 87 nM T53389 CK2Q0Y 9972086 IC50 = 1700 nM T53389 CZV48E 9972935 IC50 = 12230 nM T53389 CU3D9T 9973794 IC50 = 4100 nM T53389 C6UJ3H 9995838 IC50 = 1373 nM T53389 CYZC57 9998128 IC50 = 25 nM T53389 CPZ34K 10002593 IC50 = 117 nM T53389 CDT49B 10040459 IC50 = 24 nM T53389 C1XVD4 10049774 IC50 = 1830 nM T53389 C69VRQ 10064294 IC50 = 8 nM T53389 CU2KS9 10066538 IC50 = 630 nM T53389 CQ3G2W 10083602 IC50 = 70 nM T53389 CE79QZ 10086873 IC50 = 58 nM T53389 C1TXC3 10094943 IC50 = 5890 nM T53389 CJE5U2 10131416 IC50 = 59 nM T53389 CY8S9M 10133886 IC50 = 110 nM T53389 CZ8I7P 10150095 IC50 = 1.2 nM T53389 CVM57C 10157758 IC50 = 91 nM T53389 CJV48L 10158539 IC50 = 123 nM T53389 CU07QP 10179913 IC50 = 64 nM T53389 C30OYI 10201693 IC50 = 47 nM T53389 CSMA98 10203646 IC50 = 193 nM T53389 CQS40B 10203695 IC50 = 18 nM T53389 C9GL8R 10267580 IC50 = 25 nM T53389 CHAM93 10273926 IC50 = 110 nM T53389 CW3CN7 10274521 IC50 = 42 nM T53389 C9PRM7 10274522 IC50 = 42 nM T53389 CP3N0J 10276818 IC50 = 49 nM T53389 CHGF61 10293214 IC50 = 19 nM T53389 CY2FH3 10294883 IC50 = 30 nM T53389 CO62ML 10295106 IC50 = 40 nM T53389 CQP2T6 10321041 IC50 = 51 nM T53389 CY6C0M 10358578 IC50 = 20 nM T53389 CZV97C 10359218 IC50 = 29 nM T53389 C96UFD 10361281 IC50 = 369 nM T53389 CG65LX 10380809 IC50 = 538 nM T53389 C8X2RY 10456042 IC50 = 69 nM T53389 C3YXR2 10469233 IC50 = 2.9 nM T53389 C30DJK 10470887 IC50 = 40 nM T53389 C60HZP 10471782 IC50 = 1700 nM T53389 CDCS58 10869646 IC50 = 5800 nM T53389 C94IDS 10900715 IC50 = 2590 nM T53389 C5TJ3L 10935193 IC50 = 5100 nM T53389 C4Z9IS 10945492 IC50 = 57 nM T53389 CL3QV0 10946675 IC50 = 460 nM T53389 C2RH1W 10977011 IC50 = 3990 nM T53389 CTYB48 11033585 IC50 = 76 nM T53389 CF3LK1 11054978 IC50 = 353 nM T53389 CM6PY9 11055906 IC50 = 1760 nM T53389 CL74SR 11057468 IC50 = 400 nM T53389 CC20DE 11119216 IC50 = 150 nM T53389 CMN7K8 11150889 IC50 = 7940 nM T53389 CGV98F 11162962 IC50 = 260 nM T53389 CUL1J4 11244063 IC50 > 10000 nM T53389 CKU28N 11244510 IC50 > 10000 nM T53389 CVJ18H 11290221 IC50 = 10 nM T53389 C7M6ZR 11359080 IC50 = 30 nM T53389 CB48XU 11370662 IC50 = 1250 nM T53389 CNE51F 11439188 IC50 = 1020 nM T53389 C92QGR 11473228 IC50 = 10 nM T53389 CUJV39 11483515 IC50 > 10000 nM T53389 CGKM26 11495553 IC50 = 81 nM T53389 CC96QB 11507696 IC50 > 20000 nM T53389 C4VHE6 11508699 IC50 = 27 nM T53389 CV4UD1 11529890 IC50 = 35 nM T53389 CKJ3T4 11558948 IC50 = 115 nM T53389 CH7W3B 11588676 IC50 = 240 nM T53389 CY13AD 11594774 IC50 = 3981 nM T53389 C1FRG3 11595752 IC50 = 9333 nM T53389 C3PHJ9 11604319 IC50 = 12 nM T53389 CIM14T 11625025 IC50 = 19 nM T53389 C6LU5J 11626023 IC50 = 112 nM T53389 CGX96V 11626927 IC50 < 5011.87 nM T53389 CVUN06 11633551 IC50 = 214 nM T53389 CQ1TF6 11638261 IC50 = 59 nM T53389 CM8F3U 11675099 IC50 = 25 nM T53389 CD4Y0N 11682470 IC50 = 19 nM T53389 CH45RK 11682680 IC50 = 110 nM T53389 C1H0DJ 11716589 IC50 = 191 nM T53389 CVCU92 11717091 IC50 = 32 nM T53389 CYQ4O9 11723225 IC50 = 15 nM T53389 CWZ46B 11739564 IC50 > 10000 nM T53389 CE9MU4 11740079 IC50 = 78 nM T53389 CR14FV 11772123 IC50 = 1770 nM T53389 CG6HJ1 11780883 IC50 > 50000 nM T53389 CPF71W 11791162 IC50 = 543 nM T53389 CYE38T 11807788 IC50 = 151 nM T53389 CC09DE 11955790 IC50 = 3.2 nM T53389 C42YHI 16070117 Ki = 20 nM T53389 CWBV93 16079009 IC50 = 54.4 nM T53389 CU56EW 16664858 IC50 > 10000 nM T53389 CWO03J 16730257 IC50 > 10000 nM T53389 CM1JZ3 16730258 Ki = 54 nM T53389 C5R2QT 16730334 Ki = 11 nM T53389 C8UTH4 16730337 Ki = 19 nM T53389 CVM34Y 16730340 Ki = 78 nM T53389 CP0R2U 16730412 Ki = 111 nM T53389 CS6OA9 16730417 Ki = 640000 nM T53389 CJY8M4 16730418 Ki > 2800000 nM T53389 CT9GO8 16730419 Ki = 365 nM T53389 CW69FI 16730503 Ki = 410 nM T53389 C27IFG 16730505 Ki = 1870 nM T53389 CL59XM 16730506 Ki = 370 nM T53389 CR4IN5 16730507 IC50 > 10000 nM T53389 CMUY19 16730509 IC50 > 10000 nM T53389 C9MG5V 16730589 Ki = 190 nM T53389 C0TB2Z 16730590 Ki = 12 nM T53389 CM7E3X 16730592 Ki = 1120 nM T53389 CJET25 16730673 Ki = 24 nM T53389 CV0M6H 16730825 Ki = 35 nM T53389 C5DX2R 16730828 Ki = 78 nM T53389 CP7F1M 16730829 Ki = 5 nM T53389 C3G5MO 16730830 IC50 > 10000 nM T53389 CA6F0J 16730907 Ki > 2800000 nM T53389 CK30JX 16730909 Ki = 20 nM T53389 C75JQH 16730911 Ki = 920 nM T53389 C62OWT 16730986 Ki = 952000 nM T53389 C1Z0UG 16730990 Ki > 2800 nM T53389 CEQ53Y 16730993 Ki = 440 nM T53389 C2G3OL 16731070 Ki = 73 nM T53389 CWPZ03 16731072 Ki = 6 nM T53389 C8OPS2 16731073 Ki > 2800000 nM T53389 C39WEH 16731074 Ki = 60 nM T53389 C2MS0W 16731075 Ki = 12 nM T53389 CON47J 16731076 Ki > 2800 nM T53389 CGSE01 16731413 IC50 = 46 nM T53389 C1BXM5 16731414 IC50 = 360 nM T53389 CB4WY6 16731415 IC50 = 42 nM T53389 CH6Q2O 16731558 IC50 = 119 nM T53389 C5OI8U 16731559 IC50 = 21 nM T53389 CT40LJ 16731560 IC50 = 46 nM T53389 CF7YJ8 16731561 IC50 = 10 nM T53389 C2UPN3 16731562 IC50 = 15 nM T53389 CCRS09 16731563 IC50 = 92 nM T53389 CQZ7K4 16731722 IC50 = 24 nM T53389 CU0Q3G 16731728 IC50 = 46 nM T53389 CZ82HS 16731881 IC50 = 73 nM T53389 CQ80MT 16731882 IC50 = 47 nM T53389 CK9U7Q 16731883 IC50 = 21 nM T53389 CLHM46 16731884 IC50 = 385 nM T53389 CL5PE3 16731885 IC50 = 75 nM T53389 CE38DF 16731886 IC50 = 24 nM T53389 CBD3P7 19886439 IC50 = 1600 nM T53389 C5EFH7 21992497 IC50 = 88 nM T53389 CJQ28O 21992511 IC50 = 130 nM T53389 CO3X7S 21992575 IC50 = 48 nM T53389 C73NEC 21992630 IC50 = 74 nM T53389 CVD9T3 21992651 IC50 = 646 nM T53389 CHI3O1 21992654 IC50 = 47 nM T53389 C0QST8 21992672 IC50 = 141 nM T53389 C0QS8C 21992678 IC50 = 78 nM T53389 C5N7DG 21992681 IC50 = 343 nM T53389 C6YQV1 21992708 IC50 = 89 nM T53389 CDH32S 21992730 IC50 = 85 nM T53389 CSY41F 21992749 IC50 = 4000 nM T53389 CGJ8D2 21992811 IC50 = 24 nM T53389 C45BUO 21992812 IC50 = 100 nM T53389 CTF0Q7 21992824 IC50 = 877 nM T53389 CG03DU 21992836 IC50 = 19800 nM T53389 C7KTU1 21992839 IC50 = 9290 nM T53389 CR6F1A 21992881 IC50 > 20000 nM T53389 CBP95W 21992896 IC50 = 255 nM T53389 C6QNL9 21992913 IC50 = 71 nM T53389 CI6JQ7 23546123 IC50 = 79 nM T53389 CR7DC6 23546124 IC50 = 104 nM T53389 C2RV3U 24180608 IC50 = 296 nM T53389 C4W8IQ 24776249 IC50 = 3810 nM T53389 CQJ5Z7 24776250 IC50 = 526 nM T53389 C15UVX 24776251 IC50 = 33 nM T53389 C8G4TY 24776252 IC50 = 72 nM T53389 CF63NZ 24776253 IC50 = 1200 nM T53389 CK5Q2S 24776254 IC50 = 1100 nM T53389 CAL94V 24776255 IC50 = 4800 nM T53389 CIFD92 24776256 IC50 = 1100 nM T53389 C6NPE4 24776257 IC50 = 750 nM T53389 CV21ZF 24879059 IC50 = 16000 nM T53389 CG13IK 24879061 IC50 = 2700 nM T53389 CJ6TN2 24879098 IC50 = 4400 nM T53389 C7DU4N 24880914 IC50 = 4.3 nM T53389 CRG15B 24893986 IC50 > 1000 nM T53389 CW0MT7 24893987 IC50 > 1000 nM T53389 C4S7CP 24893988 IC50 > 1000 nM T53389 CM6XF2 25138294 Ki = 7.1 nM T53389 CDW10T 25192275 IC50 = 21 nM T53389 CF3WN9 25192277 IC50 = 22 nM T53389 CPQ31L 25195294 IC50 = 27.15 nM T53389 CA9T7Y 25195321 Ki = 15 nM T53389 C5PC2Z 25195322 Ki = 2.95 nM T53389 CSH19D 44201376 IC50 = 44 nM T53389 CN2QG1 44223357 IC50 = 33300 nM T53389 CWH5G9 44345925 IC50 = 151 nM T53389 CQVW76 44346052 IC50 = 54 nM T53389 C2UAQ1 44351275 IC50 = 61 nM T53389 CB5NF6 44408672 IC50 = 53 nM T53389 CYG2F3 44408807 IC50 = 100 nM T53389 CM54AI 44408849 IC50 = 104 nM T53389 CN4X1A 44408884 IC50 = 226 nM T53389 CF4MV9 44521014 IC50 = 13 nM T53389 CPU5Y1 44521015 IC50 = 21 nM T53389 CAT10W 44521016 IC50 = 227 nM T53389 CBF34X 44521017 IC50 = 108 nM T53389 C8Q3GP 44521018 IC50 = 107 nM T53389 CYZE89 44521019 IC50 = 7 nM T53389 C7FWV0 44521020 IC50 = 739 nM T53389 CD46PB 44521021 IC50 = 4 nM T53389 CLC0U6 44521022 IC50 = 6 nM T53389 CIN30H 44521023 IC50 = 30 nM T53389 CXFW35 44521024 IC50 = 109 nM T53389 C0V3ZN 44521025 IC50 = 12 nM T53389 CPQ14L 44521026 IC50 = 63 nM T53389 C3VRO9 44557921 IC50 > 10000 nM T53389 CIJ2Z4 44568178 IC50 > 1000 nM T53389 C29IYW 44568179 IC50 > 1000 nM T53389 CX45TP 44568180 IC50 > 1000 nM T53389 CPX96E 44568181 IC50 > 1000 nM T53389 C91EKS 44568215 IC50 > 1000 nM T53389 CTM0K2 44568298 IC50 > 1000 nM T53389 CGEA32 44568299 IC50 > 1000 nM T53389 CF16ZR 44568300 IC50 > 1000 nM T53389 C0OD3P 44568332 IC50 > 1000 nM T53389 CZT3F9 44568333 IC50 > 1000 nM T53389 CIWL70 44568334 IC50 > 1000 nM T53389 CR53DN 44568335 IC50 > 1000 nM T53389 CN43BI 44568359 IC50 > 1000 nM T53389 C4M1SH 44568360 IC50 > 1000 nM T53389 CES3O1 44568361 IC50 > 1000 nM T53389 CW52NV 44568386 IC50 > 1000 nM T53389 CSCY70 44568387 IC50 > 1000 nM T53389 CC7MB2 44568388 IC50 > 1000 nM T53389 CL95CO 44568389 IC50 > 1000 nM T53389 CZMX10 44568412 IC50 > 1000 nM T53389 CIXK10 44568413 IC50 > 1000 nM T53389 C5HRV7 44568414 IC50 > 1000 nM T53389 CCH60W 44568463 IC50 > 1000 nM T53389 C16NYL 44568698 IC50 > 1000 nM T53389 C2EXW6 44568699 IC50 > 1000 nM T53389 C56GCD 44568700 IC50 > 1000 nM T53389 C9N3UM 44568701 IC50 > 1000 nM T53389 CZMG67 44568751 IC50 > 1000 nM T53389 C0EI3M 44568752 IC50 > 1000 nM T53389 C7CH4M 44568753 IC50 > 1000 nM T53389 C03JAH 44568754 IC50 > 1000 nM T53389 CX4HV8 44570785 Ki = 2.07 nM T53389 C7A3DQ 44570786 Ki > 28000 nM T53389 CJ63ZW 44570787 Ki = 8.8 nM T53389 C9NHM1 44570788 Ki = 7.2 nM T53389 CB19GI 44571327 Ki = 19 nM T53389 CD79CQ 44571328 Ki = 53.2 nM T53389 CL5ZS4 44571329 Ki = 16.4 nM T53389 CP38YF 44571362 Ki = 15.2 nM T53389 C9TA0K 44571363 Ki = 3 nM T53389 CWF4P5 44571364 Ki = 0.7 nM T53389 CHK7O0 44571365 Ki = 0.33 nM T53389 C4OI2E 45267044 IC50 = 16 nM T53389 CC96LP 45269578 IC50 = 199 nM T53389 C2QIA8 45270417 IC50 = 93 nM T53389 CFT8P5 45271243 IC50 = 588 nM T53389 C2BXF5 45271244 IC50 = 646 nM T53389 CMT5Z2 45271247 IC50 = 3715 nM T53389 CTE15D 45272980 IC50 = 545 nM T53389 CPA4Q9 45272982 IC50 = 60 nM T53389 CCY40E 45487422 IC50 = 47 nM T53389 CN7K5Q 45487436 IC50 = 6 nM T53389 CL5D4B 45487437 IC50 = 27 nM T53389 CCA41T 45487439 IC50 = 6000 nM T53389 CXCK60 45487442 IC50 = 19500 nM T53389 CJE0F7 45487443 IC50 = 30 nM T53389 C0WY8T 45487444 IC50 = 398 nM T53389 C5O9GR 45487452 IC50 = 32 nM T53389 C7C2NK 45487453 IC50 = 50000 nM T53389 CDK6S4 45487458 IC50 = 15 nM T53389 CEGA87 45487486 IC50 = 34 nM T53389 C9LJ1W 45487500 IC50 = 40 nM T53389 C1O5PU 45487521 IC50 = 1778 nM T53389 CXO0M2 46173038 IC50 = 280 nM T53389 C8ADR2 46214481 IC50 = 3162.28 nM T53389 CH0ZR1 46214482 IC50 = 7943.28 nM T53389 C2EZU8 46214649 IC50 = 398.11 nM T53389 C5L1KH 46214650 IC50 > 10000 nM T53389 CRI6G5 46214652 IC50 = 501.19 nM T53389 CRT51W 46214653 IC50 > 10000 nM T53389 CVW21C 46215644 IC50 = 25.12 nM T53389 CZ58FY 46215814 IC50 = 1584.89 nM T53389 CO9H1K 46215816 IC50 > 10000 nM T53389 CT8G2A 46215988 IC50 > 10000 nM T53389 C28SJK 46215992 IC50 > 10000 nM T53389 C9JNT0 46216155 IC50 > 10000 nM T53389 CD96WF 46216494 IC50 = 3162.28 nM T53389 C8JQ1T 46226922 Ki = 19 nM T53389 CF91GC 46226924 Ki > 2800000 nM T53389 CH3C0F 46226927 Ki = 640 nM T53389 CIW27O 46226928 Ki > 2800000 nM T53389 C5WC9K 46871765 IC50 = 34 nM T53389 CY9SA8 46871780 IC50 = 26 nM T53389 CIP3D4 46907073 IC50 = 2250 nM T53389 C4MG6S 46907074 IC50 = 2600 nM T53389 CET36O 46907108 IC50 = 231 nM T53389 CXU48J 46907109 IC50 > 10000 nM T53389 C7Q4ZG 46907110 IC50 = 318 nM T53389 C6QLR5 46907111 IC50 > 10000 nM T53389 CWL3F7 46907143 IC50 = 131 nM T53389 C4NWF0 46907144 IC50 > 10000 nM T53389 C5ZHL8 46907145 IC50 = 255 nM T53389 CX86MP 46907146 IC50 > 10000 nM T53389 CQF0X6 46907178 IC50 = 34 nM T53389 CLT30J 46907179 IC50 = 61 nM T53389 C9PAT7 46927672 IC50 = 10 nM T53389 CRCT70 50909914 IC50 > 10000 nM T53389 C0XDI4 50909915 IC50 = 6309.57 nM T53389 CUJL92 50909916 IC50 > 10000 nM T53389 C51DKX 50909917 IC50 > 10000 nM T53389 CYD4A2 51354035 IC50 > 10000 nM T53389 CW2T3N 51354036 IC50 > 10000 nM T53389 CH8NX6 51354037 IC50 > 10000 nM T53389 CK63DI 51354327 IC50 > 10000 nM T53389 CC6PZ4 51354328 IC50 > 10000 nM T53389 C2FVX4 51354329 IC50 > 10000 nM T53389 CV06QD 51354330 IC50 > 10000 nM T53389 CR3AC1 51354331 IC50 > 10000 nM T53389 CUXD62 51354613 IC50 > 10000 nM T53389 C3G1VK 51354899 IC50 > 10000 nM T53389 CK7NP1 51354900 IC50 > 10000 nM T53389 CEDN75 51354901 IC50 > 10000 nM T53389 CB0EU1 51355190 IC50 > 10000 nM T53389 CYZ03E 51356852 IC50 = 1995.26 nM T53389 CL3S8F 51356853 IC50 = 398.11 nM T53389 C67DUF 51356854 IC50 = 501.19 nM T53389 CAU2F6 51356855 IC50 = 5011.87 nM T53389 CD07RV 51356856 IC50 > 10000 nM T53389 CFM5I7 51357137 IC50 > 10000 nM T53389 CP6R5J 51357138 IC50 = 7943.28 nM T53389 CWCJ29 51357417 IC50 > 10000 nM T53389 CS9WE1 51357418 IC50 > 10000 nM T53389 C5G7BY 51357419 IC50 > 10000 nM T53389 CBM4P9 51357696 IC50 > 10000 nM T53389 C65MXB 51357954 IC50 > 10000 nM T53389 C8HL1Q 52920793 IC50 = 22 nM T53389 C95JRW 52920794 IC50 = 25 nM T53389 C3ZK9J 52920857 IC50 = 51 nM T53389 C0U2OR 54578934 IC50 = 38 nM T53389 CDZ09I 54578935 IC50 = 13 nM T53389 CI6UG7 54578936 IC50 = 48 nM T53389 C0WM1Y 54580506 IC50 = 207 nM T53389 C4W7BZ 54580507 IC50 > 1000 nM T53389 C2AUV0 54580508 IC50 > 1000 nM T53389 CF9HP7 54580509 IC50 = 101 nM T53389 C6MXZ8 54580510 IC50 = 94 nM T53389 CCVR53 54580511 IC50 = 232 nM T53389 CRN28X 54581311 IC50 > 10000 nM T53389 CEP04I 54581525 IC50 > 1000 nM T53389 CU30TM 54582521 IC50 > 1000 nM T53389 CKAX21 54584471 IC50 > 1000 nM T53389 C0NC9L 54585425 IC50 > 1000 nM T53389 CB6XT7 54585426 IC50 > 1000 nM T53389 CA4GI9 54586383 IC50 = 75 nM T53389 C6VFC4 54586384 IC50 > 1000 nM T53389 C5MZ2T 54586385 IC50 = 88 nM T53389 CI9B8P 54670034 EC50 = 100 nM T53389 CQ2EJ5 54670128 IC50 = 15.85 nM T53389 C8JA6I 54670129 EC50 = 12.59 nM T53389 C6J7OF 54670130 EC50 = 19.95 nM T53389 C4ZBP1 54670226 EC50 = 31.62 nM T53389 C82PTD 54670693 IC50 = 7.943 nM T53389 CV9F4O 54670694 IC50 = 50.12 nM T53389 CY2M6U 54670695 IC50 = 25.12 nM T53389 C62HDF 54670783 EC50 = 31.62 nM T53389 C13LYM 54670784 IC50 = 2.512 nM T53389 C6W9QG 54671061 IC50 = 1 nM T53389 CGY8D2 54671062 EC50 = 19.95 nM T53389 C6BVG3 54671064 IC50 = 6.31 nM T53389 C0IU2E 54671255 IC50 = 2511.89 nM T53389 CQY94R 54671256 IC50 = 100 nM T53389 CEIC40 54671350 IC50 = 3.162 nM T53389 CS64EU 54764682 IC50 = 0.57 nM T53389 C3HTE0 54765510 IC50 = 5.6 nM T53389 CCZ2V9 54765512 IC50 = 6.8 nM T53389 C9M0SO 54765514 IC50 = 4.9 nM T53389 CS0HQ8 54765517 IC50 = 8.1 nM T53389 CSNW70 54765683 IC50 = 3.3 nM T53389 C6FDL2 54766012 IC50 = 13 nM T53389 C15TGK 54766018 IC50 = 13 nM T53389 C3MJ8Y 54766164 IC50 = 9 nM T53389 C7AY9N 54766165 IC50 = 17 nM T53389 CLKF74 54766166 IC50 = 9 nM T53389 CH3V8A 54766167 IC50 = 10 nM T53389 C6HX3D 54766168 IC50 = 6 nM T53389 C9E4LP 54766169 IC50 = 9 nM T53389 CL75WK 54766171 IC50 = 21 nM T53389 CD36HW 54766320 IC50 = 6 nM T53389 CL71CV 54766321 IC50 = 12 nM T53389 CG4L7Y 54766322 IC50 = 11 nM T53389 CA74KU 54766323 IC50 = 8 nM T53389 C25FDK 54766324 IC50 = 15 nM T53389 C21KGR 54766325 IC50 = 7 nM T53389 CM92AB 54766465 IC50 = 5 nM T53389 C64JAV 54766466 IC50 = 17 nM T53389 CEX96A 54766467 IC50 = 14 nM T53389 CVG4X7 54766468 IC50 = 9 nM T53389 C78SKD 54766469 IC50 = 16 nM T53389 CWV13U 54766470 IC50 = 18 nM T53389 CV9JN8 54766620 IC50 = 17 nM T53389 C5SK9R 54766621 IC50 = 14 nM T53389 CG1B5U 54766622 IC50 = 11 nM T53389 C7REA0 54766623 IC50 = 8 nM T53389 C65HJI 54766624 IC50 = 14 nM T53389 CD96AG 54766625 IC50 = 16 nM T53389 CT51IV 54766773 IC50 = 46 nM T53389 C2DIH5 54766774 IC50 = 14 nM T53389 C9W1SM 54766775 IC50 = 12 nM T53389 C56PNG 54766776 IC50 = 30 nM T53389 CJO9Y0 54766778 IC50 = 14 nM T53389 CUJ2A9 54766930 IC50 = 14 nM T53389 C7YO8F 54766931 IC50 = 48 nM T53389 C8OXL1 54766932 IC50 = 58 nM T53389 CZ5JR9 54766933 IC50 = 44 nM T53389 C7R6PT 54766934 IC50 = 14 nM T53389 C2GO1J 54767085 IC50 = 12 nM T53389 CCYX42 54767086 IC50 = 23 nM T53389 C41UWF 54767087 IC50 = 60 nM T53389 C1E2PB 54767088 IC50 = 10 nM T53389 CFB9S3 54767243 IC50 = 7 nM T53389 CUV96X 54767245 IC50 = 40 nM T53389 C7K5SJ 54767246 IC50 = 20 nM T53389 CW0GJ7 54767248 IC50 = 5 nM T53389 CN9YX4 54767249 IC50 = 30 nM T53389 CG6RC9 54767416 IC50 = 59 nM T53389 C92THY 54767417 IC50 = 13 nM T53389 CP84QJ 54767418 IC50 = 17 nM T53389 CQY04U 54767419 IC50 = 15 nM T53389 CFZ97I 54767420 IC50 = 40 nM T53389 CXO65G 54767583 IC50 = 2.9 nM T53389 CPG8U6 54767584 IC50 = 2.6 nM T53389 C5T1ZU 54767753 IC50 = 15.3 nM T53389 CS06AD 54767754 IC50 = 11 nM T53389 C3E0RV 54767755 IC50 = 22.1 nM T53389 CFL9P5 54767911 IC50 = 6.8 nM T53389 CV4I2C 54767912 IC50 = 3.1 nM T53389 CPW58S 54769997 IC50 > 1000 nM T53389 CLR3Y9 54769998 IC50 = 153 nM T53389 C1O3UI 54770205 IC50 > 1000 nM T53389 CL6FY2 54770206 IC50 = 143 nM T53389 CD6R9I 54770207 IC50 > 1000 nM T53389 C2ZV0I 54770208 IC50 = 737 nM T53389 CN4H9Z 54770209 IC50 > 1000 nM T53389 CXH87U 54770427 IC50 = 82 nM T53389 C29OBP 54770428 IC50 > 1000 nM T53389 CZ38LT 54770429 IC50 > 1000 nM T53389 C12POE 54770430 IC50 = 26 nM T53389 CSW69T 54770431 IC50 > 1000 nM T53389 C8VW1G 54770641 IC50 > 1000 nM T53389 C4U7BS 54771536 IC50 = 1.3 nM T53389 CS1R4P 54771537 IC50 = 21 nM T53389 C7G2HI 54771538 IC50 = 32 nM T53389 CG7X5S 54771759 IC50 = 9 nM T53389 CGSX68 54771760 IC50 = 55 nM T53389 C9C4VJ 54771761 IC50 = 25 nM T53389 CT8E3Q 54771762 IC50 = 11 nM T53389 C70GUO 54771763 IC50 = 78 nM T53389 CL48YQ 54771764 IC50 = 15 nM T53389 CN9QD7 56643097 IC50 > 10000 nM T53389 CHEM73 56658388 IC50 = 6430 nM T53389 CY3T2Q 56658389 IC50 = 4950 nM T53389 C7UHJ6 56658531 IC50 = 5.69 nM T53389 CZJ5F3 56661876 IC50 = 4.43 nM T53389 C7UO6H 56661877 IC50 = 3.98 nM T53389 CCGE23 56661878 IC50 = 1980 nM T53389 C18ABI 56661879 IC50 = 10 nM T53389 CIL4O7 56661886 IC50 = 95.7 nM T53389 CSMW63 56661887 IC50 = 66.8 nM T53389 CBT6M9 56661993 IC50 = 3.54 nM T53389 C6EIN3 56663574 IC50 = 77 nM T53389 CI8F9L 56665347 IC50 = 3.45 nM T53389 CO12EQ 56665348 IC50 = 4.09 nM T53389 C2XAB8 56665349 IC50 = 3680 nM T53389 CLFU05 56665484 IC50 = 4.12 nM T53389 CAG3B1 56665485 IC50 = 2.49 nM T53389 COKW25 56666809 IC50 = 68 nM T53389 C7CID9 56667031 IC50 = 32 nM T53389 C3PW1A 56668781 IC50 = 3.87 nM T53389 COMW10 56668782 IC50 = 3.3 nM T53389 CC7I6U 56668783 IC50 = 2.95 nM T53389 CS8GW6 56668784 IC50 = 5.39 nM T53389 C25RIC 56668911 IC50 = 1690 nM T53389 CEU3Z0 56668912 IC50 = 3.97 nM T53389 C7V8XC 56672248 IC50 = 2.26 nM T53389 C6KJ3F 56672249 IC50 = 2960 nM T53389 C9VI7R 56672383 IC50 = 5.08 nM T53389 CH6D7K 56675649 IC50 = 5440 nM T53389 C9YQZ5 56675650 IC50 = 3.04 nM T53389 C0OE8R 56677286 IC50 = 11 nM T53389 CPZG07 56678959 IC50 = 3220 nM T53389 CE5R8K 56678966 IC50 = 39.47 nM T53389 CH45NG 56678967 IC50 = 102 nM T53389 C6LHY3 56678968 IC50 = 85.3 nM T53389 CHJT87 56679089 IC50 = 3.98 nM T53389 C2UNH6 56679090 IC50 = 2.12 nM T53389 CSQP24 56679091 IC50 = 3810 nM T53389 CQ3N5O 56679092 IC50 = 4.37 nM T53389 CTSU71 56679674 IC50 = 2.82 nM T53389 C4X0FD 56683923 IC50 = 88 nM T53389 CJ9DL6 57400096 IC50 = 680 nM T53389 CU6QG9 57403566 IC50 = 1100 nM T53389 CKXE59 58577987 IC50 = 17.8 nM T53389 CBNJ31 58577988 IC50 = 15 nM T53389 CY7WR0 58577989 IC50 = 2.4 nM T53389 CAN79D 58577996 IC50 = 4.8 nM T53389 CTX23R 58577998 IC50 = 39 nM T53389 CIP7B1 60182373 IC50 = 3320 nM T53389 CQ6KV9 60182388 IC50 = 3960 nM T53389 C91RWL 66561650 IC50 = 13 nM T53389 C38AHD 66632799 IC50 = 47 nM T53389 CV63UL 67240318 IC50 > 10000 nM T53389 CZC9M5 67469084 IC50 = 3160 nM T53389 CF5K3C 67469574 IC50 = 19.95 nM T53389 CX2V4N 67470405 IC50 = 3.162 nM T53389 COK1L7 67470496 IC50 = 15.85 nM T53389 CE1TN8 70681473 IC50 = 69 nM T53389 C4HN7F 70682754 IC50 = 11.3 nM T53389 CGK6B1 70682755 IC50 = 9.26 nM T53389 C0V7PS 70682756 IC50 = 15.5 nM T53389 C6SDX9 70682757 IC50 = 16.9 nM T53389 CGCP65 70682763 IC50 = 22 nM T53389 CPMZ96 70683591 IC50 = 1 nM T53389 C4DKI7 70684836 IC50 = 11.2 nM T53389 CV37TR 70684847 IC50 = 22.1 nM T53389 CFS6H3 70684848 IC50 = 13.6 nM T53389 CMA38X 70686991 IC50 = 35.9 nM T53389 C87LYT 70686992 IC50 = 21.9 nM T53389 C8KBG2 70687848 IC50 = 4 nM T53389 CWXJ05 70687849 IC50 = 4 nM T53389 C8N7IV 70689057 IC50 = 10.2 nM T53389 CX2Y5O 70689058 IC50 = 19.3 nM T53389 CTH0A9 70689059 IC50 = 30.8 nM T53389 C0BIE1 70689068 IC50 = 47.7 nM T53389 C8PC1T 70689069 IC50 = 16.5 nM T53389 C0IC3J 70689070 IC50 = 25.7 nM T53389 C1DVU0 70689071 IC50 = 25.1 nM T53389 CJL0N2 70691169 IC50 = 8.75 nM T53389 CN25KI 70691183 IC50 = 15.1 nM T53389 C8X6QU 70691184 IC50 = 21.2 nM T53389 CO21AT 70692041 IC50 = 3 nM T53389 CJD7K6 70693280 IC50 = 15.8 nM T53389 CC0W1O 70693281 IC50 = 60.9 nM T53389 C7ZT3R 70695370 IC50 = 7.01 nM T53389 CY8SW6 70695371 IC50 = 24.3 nM T53389 CSUD72 70695372 IC50 = 8.92 nM T53389 CAQY83 70697381 IC50 = 11.4 nM T53389 C0I8GU 70697382 IC50 = 8.61 nM T53389 CYW19K 70697383 IC50 = 10.4 nM T53389 C91VYF 70697384 IC50 = 29.4 nM T53389 C7HS8G 70697385 IC50 = 7.43 nM T53389 C3GH1P 70697386 IC50 = 34.3 nM T53389 C3W5GQ 70697400 IC50 = 43.5 nM T53389 CKH76B 70697401 IC50 = 24.5 nM T53389 CR2U5G 70697402 IC50 = 12 nM T53389 CZ5EL7 71299325 IC50 = 240 nM T53389 C0D7VQ 71552176 IC50 = 7380 nM T53389 C5DBF6 71552177 IC50 = 8600 nM T53389 CPS30Q 71552178 IC50 = 50800 nM T53389 C30MTY 71552263 IC50 = 34500 nM T53389 C36QUN 71552267 IC50 = 4690 nM T53389 CAB7L3 72375216 IC50 = 2430 nM T53389 C08RZJ 72375217 IC50 = 990 nM T53389 CE5AB6 72375218 IC50 = 3360 nM T53389 CPFH01 72375220 IC50 = 3820 nM T53389 C3GT1R 72375222 IC50 = 2080 nM T53389 CDX54V 72375322 IC50 = 1780 nM T53389 CV6G0M 72375323 IC50 = 950 nM T53389 CL0I4M 72375324 IC50 = 240 nM T53389 CML97I 72375325 IC50 = 650 nM T53389 C9TR6D 72375326 IC50 = 800 nM T53389 CUYT59 78319219 IC50 = 18 nM T53389 C67BLK 90656196 IC50 = 85 nM T53389 C39FOS 90656197 IC50 = 78 nM T53389 C2QW6F 90656198 IC50 = 106 nM T53389 CDUS92 90656199 IC50 = 90 nM T53389 CIP5Q8 90656200 IC50 = 37 nM T53389 C3O5BS 90656201 IC50 = 57 nM T53389 C6FB0V 90656202 IC50 = 29 nM T53389 C2K0XC 90656203 IC50 = 48 nM T53389 C0CEV3 90656204 IC50 = 22 nM T53389 C31QUS 90656205 IC50 = 36 nM T53389 C4TAB6 90656206 IC50 = 27 nM T53389 CA9H7B 90656207 IC50 = 36 nM T53389 CW65FA 90656208 IC50 = 27 nM T53389 C75CEZ 91933902 IC50 = 100 nM T53389 CYX7T2 117072549 IC50 = 5140 nM T53389 CARX34 118392555 IC50 = 110 nM T53389 CA4T2K 118392556 IC50 = 4300 nM T53389 CJG8B0 118392559 IC50 = 1400 nM T53389 CN6EO5 118392561 IC50 = 82000 nM T53389 C2ZP8O 118392562 IC50 = 1910 nM T53389 C1FE4J 118392566 IC50 = 6900 nM T53389 CSXJ76 118392567 IC50 = 21000 nM T53389 CV0X1Q 118392570 IC50 = 2300 nM T53389 CM8DR2 118392571 IC50 = 95000 nM T53389 CC6K3M 118392573 IC50 = 3800 nM T53389 C5SBN1 118392585 IC50 = 26000 nM T53389 C3T8XG 118392586 IC50 = 30 nM T53389 CD3I9R 118392595 IC50 = 580 nM T53389 CQ2ZU9 118716041 IC50 = 99000 nM T53389 CDIY19 118716042 IC50 = 2800 nM T53389 CTJ0Q7 118716043 IC50 = 34800 nM T53389 C1DVT7 118716164 IC50 = 180 nM T53389 CPC0N1 118716165 IC50 = 650 nM T53389 CZD49P 118716166 IC50 = 15000 nM T53389 CA7JY6 118716167 IC50 = 28000 nM T53389 CIUJ56 118716168 IC50 = 115000 nM T53389 C87ZPY 118796358 IC50 = 3850 nM T53389 C2LD1B 121232401 IC50 = 1.9 nM T53389 CC9V0P 121411739 IC50 = 6 nM T53389 C9CV7H 121411850 IC50 = 17 nM T53389 CT9NY8 121411862 IC50 = 2 nM T53389 C09YCI 121411874 IC50 = 3 nM T53389 C9HV3A 121411904 IC50 = 2 nM T53389 CC4SD7 121411952 IC50 = 22 nM T53389 C2U3DY 121411994 IC50 = 11 nM T53389 CC2H7S 121412004 IC50 = 2 nM T53389 C7JS3L 121412028 IC50 = 5 nM T53389 CU3BI0 121412063 IC50 = 1 nM T53389 CLW35N 121412124 IC50 = 3 nM T53389 CZQO07 122196303 IC50 = 9.76 nM T53389 C7LR8Z 122196304 IC50 = 12.1 nM T53389 CGK94L 122196305 IC50 = 9.23 nM T53389 CE6UA3 122196306 IC50 = 11 nM T53389 CBXL72 122196307 IC50 = 9.81 nM T53389 C5J0HO 122196308 IC50 = 72.5 nM T53389 C6YSR2 122196309 IC50 = 41.9 nM T53389 COY82I 122196310 IC50 = 9.23 nM T53389 C0KE4Y 122196311 IC50 = 12.5 nM T53389 CMWG96 122196359 IC50 = 7.68 nM T53389 CU6L5G 122196360 IC50 = 10.8 nM T53389 CCA29B 122196361 IC50 = 13.7 nM T53389 CWB09V 122197446 IC50 = 119 nM T53389 CXD27F 122197447 IC50 = 153 nM T53389 C50GSF 122197448 IC50 = 174 nM T53389 CIHA53 122510417 IC50 = 350 nM T53389 COX7E3 122510453 Ki = 0.8 nM T53389 C26UNE 122510498 IC50 = 1.6 nM T53389 CM6Q5H 122510766 IC50 = 17 nM T53389 C0TZE4 122510927 IC50 = 0.9 nM T53389 CYE69W 126484202 IC50 = 3.9 nM T53389 CI8DF2 126484293 IC50 = 2.1 nM T53389 CUO92C 126484344 IC50 = 25 nM T53389 C8D2RG 126499376 IC50 = 1.3 nM T53389 C9MUH4 126499699 IC50 = 6.8 nM T53389 CP7DF4 126499823 IC50 = 1.7 nM T53389 CQP21J 126499825 IC50 = 1.4 nM T53389 C5K8PR 126499902 IC50 = 19 nM T53389 CWD1V7 126499983 IC50 = 62 nM T53389 CPK6O7 126537450 Ki = 0.22 nM T53389 CM42SX 126537451 Ki = 0.15 nM T53389 CYQ24M 126537506 Ki = 0.14 nM T53389 C6ZYB5 126622422 IC50 = 1.1 nM T53389 C3WGZ0 126622458 Ki = 0.14 nM T53389 C5H8LU 126677289 IC50 = 1.6 nM T53389 CI2YE9 132606873 IC50 = 7213 nM T53389 CALE74 134691232 IC50 = 1830 nM T53389 CJPO36 135223028 IC50 = 0.7 nM T53389 C5QF0M 135233366 IC50 = 90 nM T53389 C4N6OZ 135262129 IC50 = 3.4 nM T53389 CZAN82 135262182 IC50 = 2.5 nM T53389 CQ9B5Y 135262208 IC50 = 4.3 nM T53389 C6YJF9 135262382 IC50 = 4.4 nM T53389 CV72CD 135262410 IC50 = 0.96 nM T53389 C6JGV0 135421299 IC50 = 11 nM T53389 CDJY02 135442620 IC50 = 5.8 nM T53389 C52JQR 135442675 IC50 = 92 nM T53389 CCQ8J3 135454787 IC50 = 280 nM T53389 C0SCD8 135470346 IC50 = 31 nM T53389 CM9KD4 135476526 IC50 = 7.7 nM T53389 CF0V2W 135489172 IC50 = 21 nM T53389 C9P7WX 135506615 IC50 = 160 nM T53389 C5SKE8 135507480 IC50 = 8.2 nM T53389 CE5H9I 135772000 Ki = 950000 nM T53389 C3FSK4 135798077 IC50 > 10000 nM T53389 C52LCS 136042358 IC50 = 760 nM T53389 C36GMN 136042359 IC50 = 270 nM T53389 CG8K3T 136042360 IC50 = 790 nM T53389 C9C6ZD 136042361 IC50 = 2200 nM T53389 CEQS49 136042362 IC50 = 810 nM T53389 CSG49J 136042363 IC50 = 150 nM T53389 C8SQ7M 136042364 IC50 = 63 nM T53389 CYB8A1 136042365 IC50 = 420 nM T53389 C6ABH2 136042366 IC50 = 600 nM T53389 CGU89D 136042367 IC50 = 1700 nM T53389 CA21BD 136042368 IC50 = 3900 nM T53389 CHXY91 136042369 IC50 = 380 nM T53389 CYQK25 136042370 IC50 = 1700 nM T53389 CYW8A7 136042371 IC50 = 170 nM T53389 CJ7A0E 136042372 IC50 = 130 nM T53389 CHM0K9 136042373 IC50 = 730 nM T53389 CQOP23 136042374 IC50 = 1100 nM T53389 C40DGS 136042375 IC50 = 2100 nM T53389 CAU9M0 136042376 IC50 = 1200 nM T53389 CKI15V 136042377 IC50 = 1800 nM T53389 CHK91D 136042378 IC50 = 170 nM T53389 C9LFY4 136042379 IC50 = 190 nM T53389 CK4M0J 136042380 IC50 = 530 nM T53389 C5PQC6 136042381 IC50 = 130 nM T53389 CG96DL 136042382 IC50 = 30 nM T53389 CTG4C0 136042383 IC50 > 4000 nM T53389 CS06LI 136105600 IC50 = 4.5 nM T53389 C97MTA 136105601 IC50 = 8.6 nM T53389 CS3EZ4 136105602 IC50 = 8.8 nM T53389 C3NJ7H 136105610 IC50 = 9 nM T53389 CKO0J1 136105611 IC50 = 9 nM T53389 CNU9O7 136105614 IC50 = 130 nM T53389 CU5Q9E 136105618 IC50 = 8.7 nM T53389 CY1DI6 136105623 IC50 = 5.8 nM T53389 CEJ90Y 136105631 IC50 = 110 nM T53389 CLKX07 136105632 IC50 = 240 nM T53389 CQGC42 136105634 IC50 = 26 nM T53389 COW6U1 136105635 IC50 = 14 nM T53389 C0DL2V 136105638 IC50 = 74 nM T53389 C8EBH1 136105653 IC50 = 36 nM T53389 CL34QP 136105657 IC50 = 45 nM T53389 CCI0W5 136105667 IC50 = 7.2 nM T53389 CPQ27L 136105681 IC50 = 26 nM T53389 CU26FA 136105686 IC50 = 13 nM T53389 CF4N2X 136105687 IC50 = 75 nM T53389 CJIY42 136105689 IC50 = 48 nM T53389 C7H4TV 136105690 IC50 = 23 nM T53389 C1CU0R 136105692 IC50 = 79 nM T53389 CC53OK 136105695 IC50 = 12 nM T53389 CP7OS0 136105702 IC50 = 43 nM T53389 CSRQ63 136105705 IC50 = 8.1 nM T53389 C3W6YH 136105708 IC50 = 8.3 nM T53389 C41SVM 136105717 IC50 = 40 nM T53389 C0LN1A 136105739 IC50 = 7 nM T53389 CYB87Q 136105743 IC50 = 7.3 nM T53389 C7MAS4 136105752 IC50 = 37 nM T53389 CXV63U 136105756 IC50 = 17 nM T53389 C1YE3L 136105759 IC50 = 11 nM T53389 C36RBH 136226772 IC50 = 6.1 nM T53389 C19GNB 136254194 IC50 = 1 nM T53389 CE51KI 136254195 IC50 = 6 nM T53389 CSD41I 136254196 IC50 = 2 nM T53389 C72LJC 136254197 IC50 = 5 nM T53389 C0LRK5 137633390 IC50 = 25.12 nM T53389 CTQ1X7 137633948 EC50 = 100 nM T53389 C5UNM0 137636739 EC50 = 125.89 nM T53389 CUQ26A 137638483 IC50 = 25.12 nM T53389 CBEF45 137640574 EC50 = 251.19 nM T53389 CITC79 137640764 IC50 = 5.012 nM T53389 CJTK25 137641525 IC50 = 630.96 nM T53389 CE41UF 137642485 IC50 = 12.59 nM T53389 C01NKT 137646833 EC50 = 79.43 nM T53389 CINX69 137648388 EC50 = 15.85 nM T53389 CJ93LK 137648944 IC50 = 31.62 nM T53389 C85XPF 137649478 EC50 = 251.19 nM T53389 C2ES5C 137651470 IC50 = 19.95 nM T53389 CB1U4J 137652412 EC50 = 6.31 nM T53389 C4FUZ3 137652467 EC50 = 501.19 nM T53389 C2T4IJ 137652574 EC50 = 158.49 nM T53389 CW2U6K 137652663 IC50 = 7.943 nM T53389 C1UGQ6 137653247 IC50 = 7.943 nM T53389 C0N6KU 137655916 IC50 = 2.512 nM T53389 CFEU36 137656111 IC50 = 50.12 nM T53389 CR5TE3 137656175 IC50 = 316.23 nM T53389 CBG37Z 137656600 IC50 = 15.85 nM T53389 CC1UD9 137658007 IC50 = 1.995 nM T53389 CYX6S3 137658983 IC50 = 12.59 nM T53389 C57LYK 137659811 IC50 = 39.81 nM T53389 CQLH90 137661739 IC50 = 12.59 nM T53389 CPT0V7 138454752 IC50 = 18650 nM T53389 COW4V7 139582022 IC50 = 704 nM T53389 CNU4M3 145704714 IC50 > 10000 nM T53389 C6VB3O 145925651 IC50 = 25.12 nM T53389 C9RN6I 145979031 IC50 = 183 nM T53389 C5CXS9 145979203 IC50 = 181 nM T53389 C9BA4T 145979471 IC50 = 1985 nM T53389 C6OLT4 145980003 IC50 = 261 nM T53389 CS60PK 145980051 IC50 = 341 nM T53389 C82KZB 145980647 IC50 = 1413 nM T53389 CHLO29 145980744 IC50 = 5194 nM T53389 CL3IM5 145981192 IC50 = 229 nM T53389 CA34OQ 145984166 IC50 = 80 nM T53389 C6HC4V 145984387 IC50 = 2518 nM T53389 CE7K0A 145985622 IC50 = 197 nM T53389 CHYG73 145985863 IC50 = 406 nM T53389 CEA53S 145986683 IC50 = 154 nM T53389 CAMR56 145986821 IC50 = 162 nM T53389 C96GFQ 145986965 IC50 = 743 nM T53389 CJIV35 145987145 IC50 = 229 nM T53389 CC74BJ 145988090 IC50 = 147 nM T53389 C03XVG 145989616 IC50 = 612 nM T53389 CM1HY6 145990274 IC50 = 98 nM T53389 C0IO8M 145990401 IC50 = 1940 nM T53389 C08RTJ 145990712 IC50 = 548 nM T53389 C89SYI 145991013 IC50 = 517 nM T53389 CK5M9D 145991144 IC50 = 2745 nM T53389 CYQ73F 145991453 IC50 = 805 nM T53389 CU5GW9 145991466 IC50 = 1228 nM T53389 CRX7Y9 145991574 IC50 = 1288 nM T53389 CD06AN 145992193 IC50 = 97 nM T53389 CTI3L5 145992540 IC50 = 137 nM T53389 CJ4F9G 145994104 IC50 = 2008 nM T53389 CT9UE5 155510654 IC50 = 2080 nM T53389 CF2CU8 155510758 IC50 = 2910 nM T53389 C1L9IF 155510984 IC50 = 75 nM T53389 C0ZAN6 155512322 IC50 = 320 nM T53389 CUA50Q 155512496 IC50 > 5000 nM T53389 CSL73Z 155513136 EC50 = 19.95 nM T53389 C2MD1Q 155513187 IC50 > 10000 nM T53389 CQ64DF 155514482 IC50 = 1920 nM T53389 CW6C2E 155514502 IC50 > 5000 nM T53389 CY0CK6 155516843 IC50 = 15.85 nM T53389 CAL54I 155518651 EC50 = 25.12 nM T53389 CFD86N 155518907 IC50 = 25 nM T53389 CT63CU 155519108 IC50 = 3.162 nM T53389 C5N0GE 155523029 IC50 = 12.59 nM T53389 C70NHV 155523393 IC50 > 10000 nM T53389 C92VJW 155523476 IC50 = 11 nM T53389 CP4L8F 155524599 IC50 = 116 nM T53389 C5PA2F 155525040 IC50 > 5000 nM T53389 C81AHZ 155525733 IC50 > 5000 nM T53389 CPW6E9 155528043 IC50 = 312 nM T53389 CJ71GR 155528153 IC50 > 5000 nM T53389 CPEU39 155528262 IC50 = 55 nM T53389 CU9B7D 155530528 IC50 = 14 nM T53389 C3U6VQ 155532120 EC50 = 9.12 nM T53389 C9YMX3 155532969 IC50 = 66 nM T53389 C4V5SB 155533390 IC50 = 398.11 nM T53389 CR6VT8 155534625 IC50 = 3.981 nM T53389 C10DMX 155534844 IC50 = 87 nM T53389 CIF97P 155535006 EC50 = 51.29 nM T53389 CE7X0S 155536957 IC50 = 165 nM T53389 CQU0H3 155537238 IC50 = 6.31 nM T53389 C7WP5T 155537497 IC50 = 14 nM T53389 CKOC12 155537703 IC50 = 1260 nM T53389 CB6AN2 155537880 IC50 = 790 nM T53389 CY8MZ6 155538967 IC50 = 19.95 nM T53389 CBQ1O4 155539034 IC50 = 78 nM T53389 CRKI54 155540083 IC50 = 23 nM T53389 C9HOF6 155540194 IC50 = 31.62 nM T53389 C0OGZ2 155540539 IC50 = 19.95 nM T53389 C0M5HY 155541829 IC50 = 43 nM T53389 C9ML7T 155541864 IC50 = 8 nM T53389 CMK7O9 155541940 IC50 = 119 nM T53389 C4M6YT 155544005 IC50 = 63095.73 nM T53389 CMS7U8 155544549 IC50 = 30 nM T53389 CT23CQ 155544649 IC50 = 283 nM T53389 CUF13E 155546010 IC50 = 168 nM T53389 CT2S7A 155546431 IC50 = 230 nM T53389 CX9WQ7 155546694 IC50 = 21 nM T53389 CRVN92 155547073 IC50 = 42 nM T53389 CF31UZ 155547395 IC50 = 14.9 nM T53389 CL3V7C 155547885 IC50 > 5000 nM T53389 CM8E5L 155548006 IC50 = 3980 nM T53389 CRY3A2 155548898 IC50 = 3900 nM T53389 CUQ3O5 155548923 IC50 > 5000 nM T53389 C8NQ0I 155550263 IC50 = 12.59 nM T53389 C4T1BG 155550313 IC50 = 46 nM T53389 CZ9Y5A 155551667 IC50 = 30 nM T53389 C75MHC 155551790 IC50 = 17 nM T53389 C2FI6S 155552437 IC50 = 19 nM T53389 CE01LF 155553747 IC50 = 39 nM T53389 C0JV5A 155554027 EC50 = 50.12 nM T53389 CJL3D2 155555429 IC50 > 10000 nM T53389 C3JG0R 155555727 IC50 = 22 nM T53389 CY0A3R 155556360 IC50 > 5000 nM T53389 CEW5U4 155556807 IC50 = 12.59 nM T53389 CTR18O 155557674 IC50 = 3160 nM T53389 CWD8X0 155558928 IC50 > 10000 nM T53389 CV7H5S 155559048 IC50 = 320 nM T53389 CQ6P4J 155562494 IC50 = 125 nM T53389 C6UCG2 155562760 IC50 > 5000 nM T53389 C0WCO2 155563644 IC50 = 13 nM T53389 CWOE21 155564042 IC50 = 4297 nM T53389 C31ECF 155564334 IC50 = 4810 nM T53389 CK9Q5N 155564435 IC50 > 5000 nM T53389 CAZM60 155564535 EC50 = 158.49 nM T53389 CY42EB 155566265 IC50 > 10000 nM T53389 C6QY8E 155567320 IC50 = 10 nM T53389 CWE74H 155569551 IC50 = 42 nM T53389 D00JGL 6419753 IC50 = 500 nM T53389 D03ANS 9967941 IC50 = 162 nM T53389 D05BMP 11197671 IC50 = 1175 nM T53389 D05MIV 5162 IC50 = 30000 nM T53389 D05NEC 60182364 IC50 = 75 nM T53389 D06BDC 10361101 IC50 = 79 nM T53389 D06CMG 91754554 IC50 = 3000 nM T53389 D06KKN 11655119 IC50 = 3.7 nM T53389 D07ZMW 11403950 IC50 = 3540 nM T53389 D0C3AD 10202642 IC50 = 18 nM T53389 D0C7WP 4521392 Ki = 17 nM T53389 D0EU1R 46215815 IC50 > 10000 nM T53389 D0F2MP 60182389 IC50 = 178 nM T53389 D0H5CE 11231979 IC50 = 3980 nM T53389 D0H6ZP 16654987 IC50 = 12 nM T53389 D0K6YK 11676119 IC50 = 17 nM T53389 D0L0HG 766949 IC50 > 10000 nM T53389 D0PP6Y 60182393 IC50 = 10900 nM T53389 D0Q5UH 9858940 IC50 = 34.9 nM T53389 D0V3OJ 6456587 IC50 = 194 nM T53389 D0V8AC 10316032 IC50 = 35 nM T53389 D0XB4P 447966 IC50 = 40 nM T53389 D0XL7C 9796486 IC50 = 274 nM T53389 D0Y0BK 11524144 IC50 = 10000 nM T65864 D02WCI 40632 IC50 = 165400 nM T65864 D03RTS 2662 IC50 = 810 nM T65864 D09MGR 123619 IC50 = 530 nM T65864 D0AZ3C 5291 IC50 = 13700 nM T65864 D0E6XR 3062316 EC50 = 470 nM T65864 D0EG1I 9926791 IC50 > 10000 nM T65864 D0W5HK 216239 IC50 = 37.4 nM T65864 D02LBK 46883775 IC50 = 4.5 nM T65864 D02NNV 3038525 IC50 = 70 nM T65864 D02RJY 11442891 IC50 > 10000 nM T65864 D02UFQ 11620908 IC50 > 10000 nM T65864 D03HUX 49792852 IC50 > 10000 nM T65864 D03LWG 53235510 IC50 > 10000 nM T65864 D06OZJ 3008319 IC50 = 1000 nM T65864 D06TFI 10090485 IC50 = 490 nM T65864 D07EHV 44814409 IC50 > 10000 nM T65864 D07HPJ 11476171 IC50 > 10000 nM T65864 D0A5HC 45109868 IC50 = 5 nM T65864 D0C8DD 11552706 Ki = 7.943 nM T65864 D0CY1B 6420138 Ki > 10000 nM T65864 D0E3TC 44259 IC50 = 10.5 nM T65864 D0K2ZF 22049997 IC50 = 1.05 nM T65864 D0MR0B 54766013 IC50 = 1720 nM T65864 D0O0LS 25141092 IC50 > 10000 nM T65864 D0O6WV 24794418 IC50 > 2000 nM T65864 D0O6ZO 9952773 IC50 = 7.1 nM T65864 D0P1CV 46191454 IC50 > 10000 nM T65864 D0Q0AP 10409068 IC50 = 13 nM T65864 D0Q7RE 16007391 Ki > 10000 nM T65864 D0Q9UX 16718576 IC50 > 10000 nM T65864 D0R1VU 148177 IC50 = 1200 nM T65864 D0U2BH 65064 IC50 = 2210 nM T65864 D0X4MN 11597537 IC50 = 3400 nM T65864 D0LF0O 135441202 IC50 = 30970 nM T65864 D08DNZ 45102739 IC50 > 50000 nM T65864 D0W7MG 11647397 IC50 > 3000 nM T65864 D0W8BL 46868926 IC50 > 50000 nM T65864 D02MVG 11167112 IC50 = 35 nM T65864 D03KWN 11373432 IC50 = 27 nM T65864 D04WCI 16220188 IC50 = 14 nM T65864 D04YHW 11406590 IC50 = 10 nM T65864 D09ICC 5164 IC50 = 19 nM T65864 D0A9KI 9863367 IC50 = 19 nM T65864 D0F8DL 176155 IC50 = 10 nM T65864 D0H4GI 10275001 IC50 > 10000 nM T65864 D0H9KW 9578243 IC50 = 960 nM T65864 D0O7BW 12106168 IC50 = 67 nM T65864 D0T3ME 156422 Ki = 0.097 nM T65864 D0W0AM 9797240 IC50 = 38 nM T65864 CB1VW3 1400 IC50 = 1000 nM T65864 CXN25Y 5228 IC50 = 400 nM T65864 CNIW58 107905 IC50 = 1470 nM T65864 C38CSH 176920 IC50 = 39160 nM T65864 CJAF04 196969 IC50 = 250 nM T65864 C9W4UM 290221 IC50 > 15848.93 nM T65864 CIZN03 294348 IC50 = 197000 nM T65864 CCK16M 322479 IC50 = 500 nM T65864 C3NL7G 331326 IC50 = 2300 nM T65864 CS0I3K 354929 IC50 > 100000 nM T65864 C4MNG8 445840 IC50 > 10000 nM T65864 C0LET3 446816 IC50 = 794.33 nM T65864 C1YNB7 447721 IC50 = 110 nM T65864 CE76TB 447725 IC50 = 0.74 nM T65864 C3V0TX 447873 IC50 = 4 nM T65864 CB9F1O 447961 Ki > 1000 nM T65864 C1ZG2U 449087 IC50 > 10000 nM T65864 CKG76T 579429 IC50 > 15848.93 nM T65864 C0EQ6J 622378 IC50 > 15848.93 nM T65864 C2Y0RL 626628 IC50 > 15848.93 nM T65864 CXJ40G 667570 IC50 = 79 nM T65864 C18DMX 667664 IC50 = 100 nM T65864 CQ9PB5 684674 IC50 > 15848.93 nM T65864 CK89TF 766948 IC50 > 15848.93 nM T65864 CWO49I 826287 IC50 > 15848.93 nM T65864 CVY4C5 847353 IC50 > 15848.93 nM T65864 C9WV8G 936046 IC50 = 720 nM T65864 C8LFP6 969063 IC50 = 2240 nM T65864 CG0L7R 1052080 IC50 = 680 nM T65864 C9J2ZP 1076561 IC50 > 30000 nM T65864 C4XP1N 1100747 IC50 > 15848.93 nM T65864 C4R6OD 1190114 IC50 = 20400 nM T65864 C0SLP9 1489193 IC50 = 630.96 nM T65864 C92XOM 1489204 IC50 = 316.23 nM T65864 CO5K8Q 1491157 IC50 = 794.33 nM T65864 C4BR9S 1491161 IC50 = 1995.26 nM T65864 CK6QE1 1855438 IC50 = 17100 nM T65864 C1SVD2 2132479 IC50 > 100000 nM T65864 CJ1LK6 2568387 IC50 = 2300 nM T65864 CKTO92 2669062 IC50 > 10000 nM T65864 C8B0WP 2745748 IC50 = 2042 nM T65864 CVE5C7 2807754 IC50 = 220 nM T65864 CZHL80 2808202 IC50 > 50000 nM T65864 CYZ6O8 2812918 Ki = 14 nM T65864 CW6P5E 2823737 IC50 > 15848.93 nM T65864 CH9MA6 3398254 IC50 = 120 nM T65864 CVX1C3 3533224 IC50 > 25118.86 nM T65864 CU0TP2 3539049 IC50 = 25 nM T65864 CJWX69 3848929 IC50 > 100000 nM T65864 CK2QF5 4163701 IC50 = 290 nM T65864 CLN19J 4318880 IC50 = 5520 nM T65864 CKNY78 4350077 IC50 = 4740 nM T65864 CBN96T 4358655 IC50 = 4700 nM T65864 C74YTQ 4369443 IC50 = 460 nM T65864 C9SB1M 4464598 IC50 = 6.8 nM T65864 CO2SY7 4630909 IC50 = 2.6 nM T65864 CS1IU6 4912661 IC50 > 30000 nM T65864 C79ZDX 5287525 IC50 > 20000 nM T65864 CHDI45 5287728 IC50 = 6000 nM T65864 C7ZKA4 5326866 IC50 = 350 nM T65864 CR7N9O 5326869 IC50 = 340 nM T65864 C4MP5F 5327064 IC50 = 30 nM T65864 COVP86 5327065 IC50 = 30 nM T65864 C52MYD 5327893 IC50 = 488 nM T65864 CQ0ZP3 5327897 IC50 = 187 nM T65864 C7KIT4 5327898 IC50 = 105 nM T65864 CL5I2U 5330279 IC50 > 10000 nM T65864 C31FHN 5330788 IC50 = 20200 nM T65864 CDK3J0 5703619 IC50 = 11 nM T65864 CUO8A2 6467399 IC50 = 190 nM T65864 C9XM1V 6540299 IC50 = 92 nM T65864 C9WCD0 7579574 IC50 > 10000 nM T65864 CSFQ07 9549178 IC50 = 903 nM T65864 CYA76E 9798589 IC50 = 120 nM T65864 C2UE5B 9798659 IC50 = 4 nM T65864 CDKT92 9800117 IC50 = 480 nM T65864 CSH8F7 9800984 IC50 = 250 nM T65864 CNGP53 9801969 IC50 = 39 nM T65864 C1B4ZG 9802111 IC50 = 29 nM T65864 CL85DA 9803969 IC50 = 10 nM T65864 CB9ZH4 9805421 IC50 = 32 nM T65864 C20RSC 9811100 IC50 = 34 nM T65864 C9ZI4B 9814925 IC50 = 150 nM T65864 CT5M0R 9816180 IC50 = 871 nM T65864 CHV8J4 9818776 IC50 = 44 nM T65864 CMF73O 9819157 IC50 = 10 nM T65864 CP7F3K 9820742 IC50 = 130 nM T65864 CUM81R 9822690 IC50 = 21 nM T65864 C9C8YO 9824192 IC50 > 20000 nM T65864 C9LI8O 9824695 IC50 = 1320 nM T65864 C9TAL6 9826308 IC50 > 15000 nM T65864 C2L3NR 9826344 IC50 < 30 nM T65864 CRU16A 9827020 IC50 = 4.9 nM T65864 CQ3T8A 9827288 IC50 = 35 nM T65864 C5HK2A 9827930 IC50 = 30 nM T65864 COYM25 9829283 IC50 = 0.2 nM T65864 CS0XZ1 9836050 IC50 = 160 nM T65864 CV1PR2 9836051 IC50 = 150 nM T65864 C6GSZ2 9836535 IC50 = 154 nM T65864 CQR6U0 9838979 IC50 = 4300 nM T65864 CFH1J9 9839988 IC50 = 1080 nM T65864 CA6T4P 9840263 IC50 = 190 nM T65864 C83VNA 9841863 IC50 = 117 nM T65864 CXI01M 9842281 IC50 = 58 nM T65864 CKG9P8 9844525 IC50 = 88 nM T65864 CFPI31 9844683 IC50 = 2090 nM T65864 CQH58C 9844883 IC50 = 198 nM T65864 CTKV35 9845718 IC50 = 35 nM T65864 C42CVU 9846740 IC50 = 220 nM T65864 C41QWA 9857146 IC50 = 120 nM T65864 CE72OG 9857349 IC50 = 20 nM T65864 C27EAU 9858332 IC50 = 0.9 nM T65864 CP34FA 9858407 IC50 = 150 nM T65864 CRC65X 9863786 IC50 = 1 nM T65864 CEB6Y4 9863921 IC50 = 12 nM T65864 CW8V0K 9864418 Ki = 4 nM T65864 CF07OU 9864447 IC50 = 30 nM T65864 CDR82H 9865587 IC50 = 110 nM T65864 CQXO30 9867061 IC50 = 10 nM T65864 C1P8IT 9868139 IC50 = 15.7 nM T65864 CS14CX 9868339 IC50 = 90 nM T65864 CB0W3H 9869403 IC50 = 134 nM T65864 C12PKF 9871380 IC50 > 25000 nM T65864 CVK82Q 9879492 IC50 = 280 nM T65864 CFO01E 9879605 IC50 = 240 nM T65864 CJF9D2 9880709 IC50 > 15000 nM T65864 C45ENX 9883939 IC50 = 33 nM T65864 CVW95E 9884589 IC50 = 34 nM T65864 CWYF96 9884921 IC50 = 48 nM T65864 C18HKQ 9885748 IC50 = 92000 nM T65864 CJ4QV2 9885993 IC50 = 5 nM T65864 CEJ4G8 9886241 IC50 = 822 nM T65864 C5P3RD 9886349 IC50 = 6 nM T65864 CFL3S7 9887720 IC50 = 87 nM T65864 C27NAJ 9888013 IC50 = 1.4 nM T65864 C3K5OT 9889066 IC50 = 53 nM T65864 C9SU5L 9889287 IC50 = 1900 nM T65864 CU85DP 9889572 IC50 = 45 nM T65864 C8CA3X 9889622 IC50 = 6 nM T65864 CGT4L3 9889823 IC50 = 270 nM T65864 CP52JR 9889848 IC50 = 39 nM T65864 CTK3A4 9890357 IC50 = 89.13 nM T65864 CKAV96 9892864 IC50 = 70 nM T65864 CI4XL6 9900885 IC50 = 94 nM T65864 C0LPI8 9900936 IC50 = 2130 nM T65864 C7UI0P 9902305 IC50 = 6.6 nM T65864 CXTE43 9905562 IC50 = 73 nM T65864 C9XQ4I 9906682 IC50 = 7.8 nM T65864 CG47NJ 9906915 IC50 = 3020 nM T65864 C2Y3WG 9907612 IC50 > 100000 nM T65864 C3GSP5 9907874 IC50 = 180 nM T65864 CPYI29 9908316 IC50 = 3600 nM T65864 C5RE4V 9909170 IC50 = 120 nM T65864 CSOQ39 9909829 IC50 = 4100 nM T65864 CGCH17 9910722 IC50 = 300 nM T65864 CQ24AM 9922271 IC50 = 120 nM T65864 C5ZX2U 9922441 IC50 = 47.2 nM T65864 C3SAR4 9922847 IC50 = 140 nM T65864 CLM4D8 9922936 IC50 = 13 nM T65864 CIX49P 9923086 IC50 = 10.9 nM T65864 CQR6B9 9924607 IC50 = 8.8 nM T65864 CFID67 9927414 IC50 = 920 nM T65864 CTQ48P 9927432 IC50 = 500 nM T65864 CJ2MO5 9927719 IC50 = 12 nM T65864 CED2Q0 9928438 IC50 = 27 nM T65864 CX5G3A 9928616 IC50 = 18 nM T65864 CF69AC 9929037 IC50 = 160 nM T65864 C98HEM 9929101 IC50 = 100 nM T65864 CJT0A3 9929998 IC50 = 1200 nM T65864 C3V6WA 9930407 IC50 = 9 nM T65864 CGJ4M0 9931377 IC50 = 370 nM T65864 C2D5OR 9931765 IC50 = 43 nM T65864 C58QKO 9934897 IC50 = 32 nM T65864 CRZB68 9935362 IC50 = 30 nM T65864 C1T8RQ 9944397 IC50 = 160 nM T65864 C6NJ9T 9944440 IC50 = 21.6 nM T65864 CFS8T0 9944477 IC50 > 20000 nM T65864 CUGE86 9944722 IC50 = 44 nM T65864 CPLD50 9944763 IC50 = 16.6 nM T65864 CU8B0N 9944851 IC50 = 18.3 nM T65864 CK3X0O 9945364 IC50 = 32 nM T65864 CZM23F 9945595 IC50 = 17.7 nM T65864 CEWF82 9945764 IC50 = 26 nM T65864 C50UDP 9946437 IC50 = 101 nM T65864 CU0Z3A 9946911 IC50 = 50 nM T65864 C4A2SY 9946941 IC50 = 119 nM T65864 CB13JG 9947156 IC50 = 3 nM T65864 CJO47T 9948405 IC50 = 9.6 nM T65864 CYZ9K6 9949821 IC50 = 5.8 nM T65864 CB61DE 9949860 IC50 = 1200 nM T65864 C5ZVD1 9949990 IC50 = 400 nM T65864 C60EDC 9950128 IC50 = 248 nM T65864 CC50RG 9950332 IC50 = 160 nM T65864 CMO1K5 9950664 IC50 = 47 nM T65864 CS7I9D 9951380 IC50 = 290 nM T65864 C6PJ1K 9952134 IC50 > 1000 nM T65864 CKJ16G 9953051 IC50 = 130 nM T65864 CTAU02 9953522 IC50 = 105 nM T65864 C5N2DE 9953857 IC50 = 130 nM T65864 C8XVI1 9953941 IC50 = 33 nM T65864 C1YFR3 9954785 IC50 = 42 nM T65864 CBI6U7 9956363 Ki = 20 nM T65864 CJM8R9 9956715 IC50 = 1690 nM T65864 CKL51I 9957535 IC50 = 340 nM T65864 CC25KL 9957766 IC50 = 40 nM T65864 CF3S4B 9958188 IC50 = 80 nM T65864 C0V7UW 9958506 IC50 > 11000 nM T65864 CV84LA 9959427 IC50 = 30 nM T65864 C49PRD 9960569 IC50 = 50 nM T65864 CF7GU2 9965793 IC50 = 54.5 nM T65864 CDQ4T8 9966918 IC50 = 7 nM T65864 CX63PN 9967476 IC50 = 210 nM T65864 CFH9D2 9968513 IC50 = 15000 nM T65864 CMV37E 9968604 IC50 = 12.3 nM T65864 CHD79R 9969008 IC50 = 42 nM T65864 CLX82E 9974846 IC50 = 392 nM T65864 C28QAH 9975125 Ki = 130 nM T65864 C3ZR6S 9975266 IC50 = 0.7 nM T65864 C1V3EY 9982079 IC50 = 12 nM T65864 C37GXK 9983303 Ki = 1.4 nM T65864 CV8TY1 9996476 IC50 > 10000 nM T65864 CYZC57 9998128 IC50 > 10000 nM T65864 CV8I5X 9999342 IC50 = 1.8 nM T65864 CM4VP8 10001836 IC50 = 51 nM T65864 CQP98N 10002079 IC50 = 13 nM T65864 CNV50F 10002351 IC50 = 31 nM T65864 CZL05H 10002936 IC50 = 2700 nM T65864 C1W3NG 10002975 IC50 = 3.9 nM T65864 CUY0F8 10005715 IC50 > 10000 nM T65864 CYX27A 10006987 IC50 = 10 nM T65864 C5HMF0 10025752 IC50 = 6.6 nM T65864 C81WBH 10027534 IC50 = 60 nM T65864 CMZ2S8 10029735 IC50 = 224 nM T65864 CDT49B 10040459 IC50 = 250 nM T65864 CT84CR 10043924 IC50 = 7.2 nM T65864 CZQ75D 10043925 IC50 = 4.1 nM T65864 CTX6P9 10045626 IC50 = 7 nM T65864 C7YD1X 10048045 IC50 = 4 nM T65864 C6MX3C 10048112 IC50 = 40 nM T65864 CQH9A5 10050372 IC50 = 18 nM T65864 C1L6FM 10063814 Ki = 110 nM T65864 CTD1M2 10064759 IC50 = 139 nM T65864 CEKL46 10070245 IC50 = 51 nM T65864 CIW8H3 10070331 IC50 = 11 nM T65864 C2P6HN 10071040 IC50 = 752 nM T65864 C9W7GN 10072671 Ki = 17 nM T65864 CF8BY7 10072721 Ki = 6.7 nM T65864 CF1D6Y 10075240 IC50 > 10000 nM T65864 CQ3G2W 10083602 IC50 > 20000 nM T65864 C2C1BP 10089048 Ki = 10 nM T65864 C4YTF3 10089343 IC50 = 3 nM T65864 CBQL72 10089749 IC50 = 83.3 nM T65864 CBR3C2 10091017 IC50 = 20 nM T65864 CZN78J 10094158 IC50 = 1.5 nM T65864 CF1P3X 10094511 IC50 = 5100 nM T65864 C8G5RH 10095463 IC50 = 251 nM T65864 CC17JG 10098903 IC50 = 6.7 nM T65864 CVJ0G1 10113038 IC50 = 520 nM T65864 CO85BP 10114460 IC50 = 1.2 nM T65864 C37AVM 10126288 IC50 = 680 nM T65864 CV2AH1 10127604 IC50 = 6 nM T65864 CY8S9M 10133886 IC50 = 1600 nM T65864 CIF04B 10134322 IC50 = 253 nM T65864 CEHV91 10134493 IC50 = 3.1 nM T65864 C4K7UL 10134696 IC50 = 6.7 nM T65864 C7V0OB 10135552 Ki = 360 nM T65864 C6JA5L 10136387 IC50 = 2.2 nM T65864 CGI4L9 10138392 IC50 = 0.4 nM T65864 CR7UV3 10139311 IC50 = 180 nM T65864 C2S0KH 10142340 IC50 = 11 nM T65864 C9NO1X 10149689 IC50 = 46 nM T65864 CZ8I7P 10150095 IC50 = 110 nM T65864 CJF68Z 10151092 IC50 = 1900 nM T65864 CYE4T2 10151272 IC50 = 16 nM T65864 CM2DH8 10151273 IC50 = 2 nM T65864 CK50DN 10151356 IC50 = 30 nM T65864 CN0QK4 10152189 IC50 = 3.7 nM T65864 CN32WM 10155254 IC50 = 200 nM T65864 CS3ZT0 10155744 IC50 = 13 nM T65864 CKB3R5 10156282 IC50 = 482 nM T65864 CM9I0V 10156896 IC50 = 32 nM T65864 CF87VJ 10158193 IC50 = 7.9 nM T65864 C74QME 10158364 Ki = 1900 nM T65864 C69DHW 10158652 Ki = 60 nM T65864 CL7EP8 10158653 Ki = 80 nM T65864 CY09RS 10159882 Ki = 140 nM T65864 C70GNU 10160047 IC50 = 1700 nM T65864 C28CJL 10162609 Ki = 40 nM T65864 CY56HW 10163288 IC50 = 1.4 nM T65864 C29OTM 10164106 IC50 = 0.2 nM T65864 C3T6GM 10165183 IC50 = 9.1 nM T65864 CAX3U0 10166322 IC50 = 0.74 nM T65864 CR47IV 10172440 IC50 = 13 nM T65864 C28XRI 10177372 IC50 = 270 nM T65864 CTZ5J3 10177436 IC50 = 741 nM T65864 CR2PL1 10178871 IC50 = 0.9 nM T65864 C3FD4L 10178968 IC50 = 387 nM T65864 CV68DR 10179981 IC50 = 13 nM T65864 CPOB90 10181355 IC50 = 84 nM T65864 C19GNQ 10193032 IC50 = 43000 nM T65864 CCD61V 10193155 IC50 = 5300 nM T65864 CRD0W6 10194381 IC50 = 620 nM T65864 CJ4Q1N 10195333 IC50 = 160 nM T65864 C3UQ5B 10195536 IC50 = 1 nM T65864 C01IJU 10200452 IC50 = 48 nM T65864 CQU9K5 10200651 Ki = 240 nM T65864 CN3TF0 10200958 IC50 = 5.1 nM T65864 C3F1YU 10205267 IC50 = 8 nM T65864 C7QHS0 10215642 IC50 = 24 nM T65864 C4COW5 10216550 IC50 = 130 nM T65864 CWHX69 10222375 IC50 = 10 nM T65864 C40CIV 10223280 IC50 = 3 nM T65864 COSI48 10223922 IC50 = 26 nM T65864 C9PFR4 10225532 IC50 = 295 nM T65864 CCE2T5 10229750 IC50 = 17 nM T65864 C70FNL 10236731 IC50 = 900 nM T65864 CAV58E 10247424 IC50 = 9.7 nM T65864 C5TQ7X 10247543 IC50 = 1.1 nM T65864 C1I0SL 10247954 IC50 = 199.53 nM T65864 C2PW4C 10251577 IC50 = 10 nM T65864 C9GL8R 10267580 IC50 = 6720 nM T65864 C2YOJ8 10268342 IC50 = 67 nM T65864 C9HZ7F 10268386 IC50 = 947 nM T65864 CLQ25G 10269328 IC50 = 830 nM T65864 CH5K9N 10270151 IC50 = 28 nM T65864 C34FYO 10274130 IC50 = 8.1 nM T65864 CUM47C 10276213 IC50 = 2.2 nM T65864 CXU57I 10280196 IC50 = 1.1 nM T65864 CT1Y6P 10280638 IC50 = 1.1 nM T65864 CJF89L 10288541 IC50 = 2070 nM T65864 CH0N8G 10291183 IC50 = 3830 nM T65864 CU6YJ2 10291483 IC50 = 88 nM T65864 CI38KG 10295235 IC50 = 5.6 nM T65864 CS78CT 10295242 IC50 = 8.1 nM T65864 CNL21U 10295475 Ki = 100 nM T65864 C20HDW 10295799 IC50 = 8 nM T65864 C7SFI1 10296883 IC50 > 10000 nM T65864 CV1WZ5 10301047 IC50 = 22 nM T65864 CFV1D3 10301843 IC50 = 37 nM T65864 C5EI2W 10302380 IC50 = 34 nM T65864 CB59MP 10310219 IC50 = 8.7 nM T65864 CPU1Q8 10310740 IC50 = 10 nM T65864 C5LM2F 10316101 IC50 = 8.8 nM T65864 CPS9U3 10319232 IC50 > 10000 nM T65864 CW3AH9 10319451 IC50 = 94 nM T65864 CC2ZT0 10319912 IC50 = 7.1 nM T65864 CWYD38 10321190 IC50 = 7.413 nM T65864 C3G5OU 10337188 IC50 = 24 nM T65864 CUN52O 10345191 IC50 = 34 nM T65864 CFTS09 10346232 IC50 = 14.5 nM T65864 CY6C0M 10358578 IC50 > 15000 nM T65864 C5QE2W 10359123 IC50 = 58 nM T65864 CHA13D 10361020 IC50 = 11.1 nM T65864 C96UFD 10361281 IC50 = 510 nM T65864 CFL5O8 10364826 IC50 = 40 nM T65864 CZ74PO 10365336 IC50 = 2240 nM T65864 CDS29Z 10366675 IC50 = 108 nM T65864 C03UPC 10366721 IC50 < 30 nM T65864 CG65LX 10380809 IC50 = 280 nM T65864 C7BUP1 10382478 IC50 = 3.5 nM T65864 CKU31J 10383002 IC50 = 730 nM T65864 C6HM7N 10384508 IC50 = 2.3 nM T65864 C4FBG5 10386963 IC50 = 128 nM T65864 CVER47 10388586 IC50 = 79 nM T65864 CNL2U9 10389147 IC50 = 3 nM T65864 CU4R9M 10413666 IC50 = 330 nM T65864 C7HBP6 10429593 IC50 > 10000 nM T65864 CSO2J3 10431035 IC50 = 14 nM T65864 CC1A0N 10436869 IC50 = 26.1 nM T65864 CQ4C7Y 10450926 IC50 = 188 nM T65864 CSAZ29 10454329 IC50 = 133 nM T65864 CY9DS7 10458235 IC50 = 135 nM T65864 CS57UV 10458352 IC50 = 34.7 nM T65864 C3YXR2 10469233 IC50 = 78 nM T65864 CWY7D1 10469531 Ki = 87 nM T65864 C30DJK 10470887 IC50 > 10000 nM T65864 C2WQ8M 10473563 IC50 = 3.2 nM T65864 CG5R0N 10475624 IC50 = 18 nM T65864 C6ZEV1 10475737 IC50 = 58 nM T65864 CL5GO8 10477230 IC50 = 27 nM T65864 C68BCP 10478416 IC50 = 8 nM T65864 CRX6F0 10479082 Ki = 1.7 nM T65864 CB47LY 10847715 IC50 > 15848.93 nM T65864 CW17GM 10862277 IC50 = 1970 nM T65864 C8DW2Z 10862355 IC50 = 65 nM T65864 C6K2YS 10862784 IC50 = 2100 nM T65864 C6T8MO 10872508 IC50 = 5 nM T65864 CD8P0C 10873194 IC50 = 12000 nM T65864 C73VMQ 10874554 IC50 = 3800 nM T65864 CKG4N2 10883362 IC50 = 5700 nM T65864 CG5QT8 10884047 IC50 = 2300 nM T65864 C94IDS 10900715 IC50 = 6800 nM T65864 C5KNF9 10915062 IC50 = 440 nM T65864 C4LR6A 10928000 IC50 = 3800 nM T65864 CR85ZB 10935149 IC50 = 86 nM T65864 CT9H5W 10937337 IC50 = 1 nM T65864 C1NAT9 10938334 IC50 = 50 nM T65864 C4Z9IS 10945492 IC50 > 20000 nM T65864 CJY80W 10948417 IC50 = 35000 nM T65864 CO49ZL 10948887 IC50 = 258 nM T65864 CI3HC4 10957154 IC50 = 1800 nM T65864 C4Z8GP 10959756 IC50 = 3 nM T65864 CGI56J 10970903 IC50 = 100 nM T65864 C2LEG7 10972432 IC50 = 750 nM T65864 CA53TB 10972838 IC50 = 2300 nM T65864 C2RH1W 10977011 IC50 > 20000 nM T65864 C9GX6I 10980521 IC50 = 172 nM T65864 CNYW82 10980912 IC50 = 23600 nM T65864 CMG97R 10992192 IC50 = 437 nM T65864 CN5UP8 11001230 IC50 = 3300 nM T65864 C76JPU 11004637 IC50 = 1500 nM T65864 C5UZ8K 11011691 IC50 = 3100 nM T65864 CL3M7B 11011717 IC50 = 53 nM T65864 CS96HY 11012564 IC50 = 24 nM T65864 CEDQ13 11014525 IC50 = 217 nM T65864 CKJ29N 11024350 IC50 = 690 nM T65864 CTYB48 11033585 IC50 = 1300 nM T65864 C5WG1I 11035416 IC50 = 21 nM T65864 CTVO34 11048442 IC50 = 3400 nM T65864 CF3LK1 11054978 IC50 = 400 nM T65864 CM6PY9 11055906 IC50 = 2300 nM T65864 CA7C3T 11090422 IC50 = 139 nM T65864 CZP29I 11091452 IC50 = 1400 nM T65864 C7EH8X 11098241 IC50 = 895 nM T65864 COE34F 11103319 IC50 = 12 nM T65864 CC20DE 11119216 IC50 = 7700 nM T65864 C5X2ZF 11120768 IC50 = 1040 nM T65864 CS1Q4I 11121456 IC50 = 813 nM T65864 C3P0VX 11133737 IC50 = 8.5 nM T65864 CL7W0D 11154535 IC50 = 1850 nM T65864 C6D9HX 11155124 IC50 = 65 nM T65864 CG0M6Q 11155286 IC50 = 2029 nM T65864 CN4QP1 11157369 IC50 = 4.4 nM T65864 CJ93PH 11157370 IC50 = 4.4 nM T65864 CSM49E 11177303 IC50 = 42 nM T65864 CK4DN6 11178413 IC50 = 120 nM T65864 C2OR0F 11179277 IC50 = 4.8 nM T65864 C3ZOG2 11184891 IC50 = 193 nM T65864 CH3P1J 11186612 IC50 = 4.5 nM T65864 C91FSN 11188019 IC50 = 2 nM T65864 CLSG31 11188488 IC50 = 1600 nM T65864 C9R6ZP 11188782 IC50 = 150 nM T65864 CXK47R 11188783 IC50 = 8692 nM T65864 CU3O4M 11192376 IC50 = 57 nM T65864 C0Y8TX 11192751 IC50 > 10000 nM T65864 CEUR60 11192985 IC50 > 10000 nM T65864 CA2E1S 11201072 IC50 = 666 nM T65864 CD1U6L 11202500 IC50 = 125 nM T65864 C38UDX 11203064 IC50 = 2512 nM T65864 C9M4JX 11203238 IC50 = 4.7 nM T65864 CB06ZF 11204217 IC50 > 10000 nM T65864 CUG6B9 11208869 IC50 = 574 nM T65864 CY02IT 11209289 IC50 = 143 nM T65864 CEJ6F2 11214762 IC50 > 10000 nM T65864 C25EQP 11215012 IC50 = 1306 nM T65864 CMH0D3 11220119 Ki > 2500 nM T65864 C6TF5U 11224170 IC50 = 4099 nM T65864 C8Q0KL 11224214 IC50 = 54 nM T65864 C5LM1P 11224552 IC50 = 9.9 nM T65864 C06ZRN 11224854 IC50 = 3732 nM T65864 CV91QN 11225063 IC50 = 2.7 nM T65864 CZ78SL 11226823 IC50 > 10000 nM T65864 CPN9K8 11234551 IC50 = 110 nM T65864 C2W5RC 11235063 IC50 = 4.1 nM T65864 CQY90F 11236166 IC50 = 4570.88 nM T65864 CZ06EN 11244981 IC50 = 22 nM T65864 CWD28N 11256035 IC50 = 3.5 nM T65864 CCD5V8 11256129 IC50 = 1550 nM T65864 C1I0TQ 11257459 IC50 = 63 nM T65864 CAR3X1 11259005 IC50 = 2 nM T65864 CCED24 11260440 IC50 = 5849 nM T65864 CC2L8U 11268003 IC50 = 2.3 nM T65864 C5HRC0 11268703 IC50 = 9900 nM T65864 CYX96C 11269935 IC50 = 671 nM T65864 CEA01Q 11270757 IC50 = 190 nM T65864 CT0Z5E 11271166 IC50 = 1220 nM T65864 CR0L9N 11281388 IC50 = 20.7 nM T65864 CX3B5O 11285013 IC50 > 10000 nM T65864 CQ4DE0 11293575 IC50 = 530 nM T65864 CE2AJ5 11304134 IC50 = 110 nM T65864 CJS9C0 11304851 IC50 = 25000 nM T65864 CUQK84 11305782 IC50 = 22 nM T65864 CP7M2V 11307841 IC50 = 4435 nM T65864 C43RFW 11315961 IC50 = 205 nM T65864 CI6EC5 11324104 IC50 = 29 nM T65864 C95WQP 11326501 IC50 = 4.2 nM T65864 CCI3X6 11326593 IC50 = 4.2 nM T65864 CU5P8C 11331007 IC50 > 10000 nM T65864 C6AW3V 11339038 IC50 = 431 nM T65864 C7L1PX 11348753 IC50 = 5 nM T65864 C25JGP 11353237 IC50 > 10000 nM T65864 CTN8Y9 11353960 IC50 > 10000 nM T65864 C54CWH 11364404 IC50 = 5.5 nM T65864 CGN8P2 11365768 IC50 > 10000 nM T65864 CGW8R0 11366073 IC50 = 19.9 nM T65864 C9DYG3 11373706 IC50 = 7290 nM T65864 CPZ27G 11375263 IC50 = 250 nM T65864 C56ZGC 11376142 IC50 = 310 nM T65864 CX9UC1 11376336 IC50 = 18 nM T65864 CT6Y9W 11376799 IC50 > 10000 nM T65864 CRB0Q8 11377434 IC50 = 22.8 nM T65864 CEAR81 11381572 IC50 = 3.2 nM T65864 C9N0VD 11385711 IC50 = 250 nM T65864 CWX1M2 11387338 IC50 = 2377 nM T65864 CG18UN 11394491 IC50 = 54 nM T65864 CG9Y8F 11395429 IC50 = 5.4 nM T65864 C3JI9L 11396732 IC50 = 1260 nM T65864 CBV6F9 11396845 IC50 = 1110 nM T65864 CH7KE1 11397096 IC50 = 2670 nM T65864 CT3VP7 11398307 IC50 = 1650 nM T65864 C7F6BS 11407773 IC50 = 8479 nM T65864 C8S1PW 11409925 IC50 = 460 nM T65864 CIA75B 11410766 IC50 = 4.3 nM T65864 C5URB2 11410894 IC50 = 1420 nM T65864 C9HVR8 11411011 IC50 = 15.3 nM T65864 CYW65I 11417763 IC50 = 3.8 nM T65864 C52RJE 11418329 IC50 = 14 nM T65864 CR2MX3 11418521 IC50 = 2409 nM T65864 C0WT1L 11421331 IC50 = 150 nM T65864 C5O1RM 11421633 IC50 = 7500 nM T65864 CI5W8G 11421730 IC50 = 190 nM T65864 C0APW4 11422034 IC50 = 4800 nM T65864 C71PYD 11427975 IC50 = 4 nM T65864 CB4E7Q 11430712 IC50 = 1200 nM T65864 C5NU1W 11430933 IC50 = 1343 nM T65864 CTUM34 11431185 IC50 = 270 nM T65864 CC8U3S 11438287 Ki = 97 nM T65864 C3AS8V 11439407 IC50 = 3.4 nM T65864 C84SZX 11442171 IC50 = 110 nM T65864 C4H7QN 11444535 IC50 = 71 nM T65864 CKM8E6 11444953 IC50 > 10000 nM T65864 CFR80G 11454030 IC50 = 158 nM T65864 CJC95A 11454205 IC50 = 44 nM T65864 C1JKY5 11454412 IC50 = 1360 nM T65864 C0OAI4 11455262 IC50 = 2236 nM T65864 CU50OG 11455909 IC50 = 4300 nM T65864 C9WN4P 11463583 IC50 = 313 nM T65864 CP2R6S 11465681 IC50 = 345 nM T65864 C2MEI7 11467224 IC50 > 10000 nM T65864 C2VD6T 11472619 IC50 = 4.1 nM T65864 CYES96 11473981 IC50 = 811 nM T65864 CDOF16 11484790 IC50 = 2 nM T65864 C4PJL3 11484931 Ki = 1100 nM T65864 C19GUZ 11486266 IC50 = 5900 nM T65864 CIG0B7 11488218 IC50 = 6279 nM T65864 C29SHG 11489361 IC50 = 70 nM T65864 CLR19A 11489559 IC50 > 10000 nM T65864 CV5I3W 11490693 IC50 = 15.9 nM T65864 C7K1CO 11495230 IC50 = 39.9 nM T65864 C28NDF 11496473 IC50 = 240 nM T65864 CY49JK 11502177 IC50 = 1250 nM T65864 CO1NE9 11502288 IC50 = 31 nM T65864 CN59QW 11502801 IC50 = 2.73 nM T65864 CP37MN 11508284 IC50 = 4040 nM T65864 CHT83Z 11509206 IC50 = 201 nM T65864 CU2OF8 11510392 IC50 = 109 nM T65864 CM7D5Q 11511121 IC50 = 250 nM T65864 CI58XU 11511369 IC50 = 855 nM T65864 C8AY3B 11518031 IC50 = 12 nM T65864 C7A4GY 11524665 IC50 = 2.2 nM T65864 CBH9Z0 11529613 IC50 = 2780 nM T65864 CGC8Z2 11529647 IC50 > 56000 nM T65864 C5T9ZA 11530816 IC50 = 9540 nM T65864 C0VB6Q 11531118 IC50 = 31 nM T65864 CX27YT 11531595 IC50 = 360 nM T65864 CN16AM 11532502 IC50 = 12 nM T65864 CF0EA3 11533187 IC50 = 48 nM T65864 C5ZWR1 11538523 IC50 = 181 nM T65864 CI1C7D 11538813 IC50 = 7.8 nM T65864 CD3UE0 11540078 IC50 = 5700 nM T65864 CU27LT 11540303 IC50 = 2300 nM T65864 CNM69V 11540339 IC50 = 120 nM T65864 C2NLT0 11545778 IC50 = 210 nM T65864 CB6Z8C 11545890 IC50 = 3130 nM T65864 CCZ36R 11546418 IC50 > 5000 nM T65864 C9MFI3 11546637 IC50 = 4.4 nM T65864 CR25AP 11546709 IC50 = 539 nM T65864 CT3BY8 11546846 IC50 = 42 nM T65864 C0AZ2Q 11547059 IC50 = 2000 nM T65864 C2I4PQ 11547192 IC50 = 12 nM T65864 CN3KT0 11547541 IC50 = 10 nM T65864 CPH9B0 11551077 IC50 = 53 nM T65864 CWVP14 11551783 IC50 > 10000 nM T65864 CIRM93 11552798 IC50 = 520 nM T65864 CP3E5U 11554076 IC50 = 4.677 nM T65864 C5Z1TJ 11554246 IC50 = 36 nM T65864 CX8JT7 11554302 IC50 = 50 nM T65864 C89KGM 11554629 IC50 = 220 nM T65864 C8WD4A 11559464 IC50 > 10000 nM T65864 C5OZY0 11561357 IC50 = 1410 nM T65864 C2ID6H 11561850 IC50 = 10000 nM T65864 CA1WC9 11565393 IC50 = 100 nM T65864 CQ1RA3 11565394 IC50 = 6700 nM T65864 CNP2U5 11566683 IC50 = 520 nM T65864 CY0T8J 11567867 IC50 = 2000 nM T65864 C6B9MN 11568399 IC50 = 212 nM T65864 CC82HT 11568587 IC50 = 30 nM T65864 CMK6Z2 11569298 IC50 = 83 nM T65864 CFV89X 11569316 IC50 = 130 nM T65864 C8BD7L 11575255 IC50 > 10000 nM T65864 C2BVO6 11575331 IC50 = 6080 nM T65864 C1AX0F 11575475 IC50 = 718 nM T65864 C9U5RT 11576179 IC50 = 22 nM T65864 C1WU0N 11580175 IC50 = 530 nM T65864 CCS2N9 11583248 IC50 = 25 nM T65864 C1FBE5 11590182 IC50 = 135 nM T65864 CDG0T3 11590305 IC50 > 5000 nM T65864 C57TVC 11591147 IC50 = 367 nM T65864 CC03QG 11591157 IC50 = 6400 nM T65864 C37OKW 11591429 IC50 = 18 nM T65864 COL5U0 11591602 IC50 = 3160 nM T65864 C6SW9P 11594806 IC50 > 30000 nM T65864 CD6KY4 11596384 IC50 = 293 nM T65864 C0MBN9 11596656 IC50 = 22300 nM T65864 C8V4NP 11597359 IC50 = 20.5 nM T65864 C3XJY4 11601759 IC50 = 640 nM T65864 CJV48I 11602903 IC50 = 170 nM T65864 CA3J8I 11604225 IC50 = 176 nM T65864 C1I3UJ 11605092 IC50 = 18 nM T65864 CK35WT 11605202 IC50 > 10000 nM T65864 CA4J6X 11605249 IC50 = 1200 nM T65864 C1HV4Y 11605487 IC50 = 110 nM T65864 C4IMG2 11611340 IC50 > 1000 nM T65864 C6O3BN 11611482 IC50 = 30 nM T65864 CINC08 11612573 IC50 = 130 nM T65864 CHA59Z 11618088 IC50 = 40 nM T65864 C8Q4LX 11618535 IC50 = 130 nM T65864 C9DJ6H 11619376 IC50 = 46.5 nM T65864 CG2PW5 11619378 IC50 = 91 nM T65864 CV4Z6T 11619786 IC50 = 5 nM T65864 C5B3XJ 11620410 IC50 > 40000 nM T65864 C5D1TG 11624479 IC50 = 30 nM T65864 CA2OB4 11624640 IC50 = 1280 nM T65864 C31ZDN 11625524 IC50 = 5.48 nM T65864 CHB3F2 11626055 IC50 = 10.9 nM T65864 CSM62L 11626920 IC50 = 5 nM T65864 CGX96V 11626927 IC50 > 15848.93 nM T65864 C41IYQ 11626968 IC50 = 900 nM T65864 CPV1H5 11630444 IC50 > 100000 nM T65864 CYS76K 11632113 IC50 = 1200 nM T65864 CC36RU 11633476 IC50 = 86 nM T65864 CRSB81 11634170 IC50 = 3500 nM T65864 CQE08U 11634475 IC50 = 76 nM T65864 COLF16 11639342 IC50 = 1072 nM T65864 CGE4R2 11640131 IC50 = 1040 nM T65864 CI5J7G 11640137 IC50 = 6.88 nM T65864 CRP81Z 11641039 IC50 = 2000 nM T65864 CKC09N 11643997 IC50 > 667000 nM T65864 C4GTZ8 11645322 IC50 > 20000 nM T65864 C56VKX 11646635 IC50 = 241 nM T65864 CJ6T4Y 11646914 IC50 = 60.8 nM T65864 CW6CA5 11654334 IC50 = 3.62 nM T65864 CWLZ32 11655437 IC50 = 1700 nM T65864 C61XCD 11660643 IC50 = 6590 nM T65864 C15XRN 11663096 IC50 = 15 nM T65864 C3LH7E 11673569 IC50 = 2860 nM T65864 C2XZE7 11674063 IC50 = 240 nM T65864 C1LV6N 11675697 IC50 = 110 nM T65864 CKI36N 11675748 IC50 = 60 nM T65864 C82RWT 11677752 IC50 = 110 nM T65864 C7T9ES 11681588 IC50 = 190 nM T65864 C1AIW6 11682474 IC50 = 13 nM T65864 CJ9KN7 11683817 IC50 = 12 nM T65864 CU53MJ 11685293 IC50 = 1.7 nM T65864 C7ZE6M 11689340 IC50 = 40 nM T65864 C1YP9W 11690379 IC50 = 5.4 nM T65864 CU0E8O 11690457 Ki > 4000 nM T65864 CAF2I3 11691493 IC50 = 79 nM T65864 C10HDB 11697337 IC50 = 120 nM T65864 CQ2VU1 11697345 IC50 = 1740 nM T65864 C5N4MU 11698246 IC50 = 520 nM T65864 CY9S4V 11698813 IC50 = 6 nM T65864 CS5ZC1 11702482 IC50 = 4.8 nM T65864 CLJR20 11702517 IC50 = 9680 nM T65864 CV29PN 11703664 IC50 = 7420 nM T65864 CM1B8O 11705179 IC50 = 16000 nM T65864 CB0AP2 11705863 Ki > 4000 nM T65864 CJ37CH 11710028 IC50 = 160 nM T65864 C0OHA6 11711836 IC50 = 1.8 nM T65864 C1N3YZ 11716060 IC50 = 510 nM T65864 CYDU57 11716469 IC50 = 8380 nM T65864 CZ2PC3 11717079 IC50 = 12.3 nM T65864 C7HOZ4 11718141 IC50 = 4640 nM T65864 CLJ18D 11719217 IC50 = 122 nM T65864 CVC2S4 11722798 IC50 > 10000 nM T65864 C9S5JI 11732012 IC50 = 2900 nM T65864 CQ4MV7 11737779 IC50 = 145 nM T65864 C3AKG6 11744373 IC50 = 11 nM T65864 CBQP05 11749046 IC50 = 5080 nM T65864 CN8S1E 11752715 IC50 > 10000 nM T65864 C52ZHW 11752855 IC50 = 2001 nM T65864 CVSO90 11753013 IC50 = 4.5 nM T65864 CXQO43 11753341 IC50 = 4974 nM T65864 C2N9IP 11767594 IC50 = 1200 nM T65864 CPU1B6 11785271 IC50 > 10000 nM T65864 CL87KR 11785748 IC50 > 10000 nM T65864 C7D1GP 11785826 IC50 = 9501 nM T65864 CZ58LK 11786348 IC50 > 10000 nM T65864 CD5SM9 11786421 IC50 = 52 nM T65864 CYZ8V2 11786594 IC50 = 38 nM T65864 CPF71W 11791162 IC50 > 20000 nM T65864 CYE38T 11807788 IC50 > 20000 nM T65864 C5LT9N 11809327 IC50 = 68 nM T65864 CO7RA4 11814282 IC50 = 1200 nM T65864 CX71IE 11822822 IC50 = 98 nM T65864 C38XYS 11825589 IC50 = 185 nM T65864 CCT2E5 11833097 IC50 = 6.5 nM T65864 CFHX82 11837140 IC50 > 100000 nM T65864 CCI6R5 11842847 IC50 = 1200 nM T65864 CMO6N4 11842849 IC50 = 1800 nM T65864 C9HT7B 11842850 IC50 = 8000 nM T65864 CP6KY2 11843009 IC50 = 430 nM T65864 C8FHK9 11843010 IC50 = 2100 nM T65864 C7D6MQ 11843012 IC50 = 1200 nM T65864 C4T2WC 11843013 IC50 = 2300 nM T65864 CS36BH 11843159 IC50 = 530 nM T65864 C7DU6T 11843160 IC50 = 6800 nM T65864 CH6W3V 11844349 IC50 = 160 nM T65864 CI15NA 11844350 IC50 = 320 nM T65864 CUL2C8 11844485 IC50 = 740 nM T65864 C96ORQ 11844486 IC50 = 440 nM T65864 C4SK3L 11844487 IC50 = 1000 nM T65864 C6KF8Z 11844488 IC50 = 2100 nM T65864 C9ECK3 11844489 IC50 = 180 nM T65864 C83YRX 11844616 IC50 = 1300 nM T65864 CV24WL 11844764 IC50 = 420 nM T65864 C9JT4S 11847343 IC50 > 10000 nM T65864 CAZS08 11848309 IC50 = 0.6 nM T65864 C43IVN 11848567 IC50 = 2 nM T65864 C9LAY8 11848825 IC50 = 1.1 nM T65864 CI4F2L 11854236 IC50 = 1 nM T65864 C89FTX 11854237 IC50 = 2 nM T65864 CA2LF8 11947957 IC50 = 1 nM T65864 C27ALB 11955788 IC50 = 100 nM T65864 CWM32N 11957412 IC50 = 9 nM T65864 CW6XN7 11962205 IC50 = 3060 nM T65864 C0R7ZI 11962712 IC50 = 196 nM T65864 CH5T7F 11962713 IC50 = 300 nM T65864 C40DWV 11962714 IC50 > 5000 nM T65864 CS71YJ 11962715 IC50 = 1316 nM T65864 CGV83D 11962718 IC50 = 1219 nM T65864 C1YDM5 11962719 IC50 > 5000 nM T65864 CN0B6Q 11962793 IC50 = 239 nM T65864 CAN64P 11962794 IC50 = 3021 nM T65864 CUE29A 11962795 IC50 > 5000 nM T65864 C0YHS3 11962796 IC50 = 1171 nM T65864 CY0EX4 11977143 IC50 = 1090 nM T65864 C8E4TS 11992146 IC50 = 87000 nM T65864 CVW2E9 11996858 IC50 = 8.128 nM T65864 CJ9O1A 12000612 IC50 = 20 nM T65864 CTP7S1 12084786 IC50 = 53 nM T65864 C1S4UX 12113733 IC50 = 285 nM T65864 CY7F1N 12150537 IC50 = 390 nM T65864 CXU6M2 12310041 IC50 = 252000 nM T65864 C0XE2H 12967031 IC50 = 1400 nM T65864 C7N4DA 12967032 IC50 = 420 nM T65864 CAVB53 12967033 IC50 = 420 nM T65864 CR91OX 12967034 IC50 = 80 nM T65864 C86PGJ 12967035 IC50 = 4740 nM T65864 CIQ7M6 14198571 IC50 > 15848.93 nM T65864 C3YRU7 15295578 IC50 > 50000 nM T65864 CX8Z9K 15407403 IC50 = 33 nM T65864 C8WKH7 15513074 IC50 = 16.5 nM T65864 CBA4X0 15513101 IC50 = 97.4 nM T65864 CMAI91 15547874 IC50 = 36 nM T65864 CGV5T1 15547875 IC50 = 370 nM T65864 CLJ9D2 15547876 IC50 = 120 nM T65864 CBMG59 15547877 IC50 = 1100 nM T65864 COQ93C 15547878 IC50 = 290 nM T65864 CVO3X1 15547880 IC50 = 120 nM T65864 CH19QA 15680125 IC50 > 15848.93 nM T65864 C0OQ5J 15872094 IC50 > 20000 nM T65864 C1C6FX 15872095 IC50 = 15000 nM T65864 C6EQ7J 15872096 IC50 = 20000 nM T65864 C70YDR 15872098 IC50 = 370 nM T65864 C7VF9T 15872388 IC50 = 19 nM T65864 C47UOV 15872390 IC50 = 317 nM T65864 C7LD2G 15872391 IC50 = 177 nM T65864 C4CDK1 15872392 IC50 = 14.13 nM T65864 CQZ92D 15872393 IC50 = 12 nM T65864 C7DEG6 15872398 IC50 = 18.7 nM T65864 C4EN7J 15872399 IC50 = 60 nM T65864 CN0QB9 15872400 IC50 = 128.82 nM T65864 C5I0MB 15872401 IC50 = 20 nM T65864 CBU15L 15872403 IC50 = 22.91 nM T65864 CTXY45 15872404 IC50 = 95.5 nM T65864 CPQ31T 15872405 IC50 = 13 nM T65864 CTK30G 15872406 IC50 = 25 nM T65864 CU1XR0 15872407 IC50 = 132 nM T65864 CAUI95 15872408 IC50 = 208.93 nM T65864 C4P6MA 15872409 IC50 = 645.65 nM T65864 CZ1H2L 15887011 IC50 = 34.3 nM T65864 C8HZ1V 15887012 IC50 = 15.14 nM T65864 C51ARC 15887024 IC50 = 56.23 nM T65864 C9RQN8 15950748 IC50 = 14 nM T65864 CZ6B2Y 15951509 IC50 = 83 nM T65864 CWN98Z 15953778 IC50 = 0.51 nM T65864 CEB0A6 15953837 IC50 = 23 nM T65864 CAV34S 15987404 IC50 = 3.2 nM T65864 CW02NJ 15987405 IC50 = 17 nM T65864 CBF4X2 15991561 IC50 > 15848.93 nM T65864 CSK90Y 15991573 IC50 = 6 nM T65864 CPNW35 15991575 IC50 = 76 nM T65864 C8TW5P 16007071 IC50 = 28 nM T65864 C09OWB 16015442 IC50 = 14445 nM T65864 CA1FM3 16043321 IC50 = 0.6 nM T65864 C9TU1O 16046126 IC50 > 1000 nM T65864 CP0M4R 16048965 IC50 = 42.7 nM T65864 CL67VN 16049878 IC50 = 5 nM T65864 CWBV93 16079009 IC50 = 594 nM T65864 CKV4G1 16079040 IC50 = 35000 nM T65864 C3ZV2X 16086076 IC50 = 9 nM T65864 C0SO7D 16086077 IC50 = 2 nM T65864 C0WU9I 16086078 IC50 = 2 nM T65864 CVE6C8 16086088 IC50 = 2 nM T65864 CH1R8K 16086091 IC50 = 0.9 nM T65864 CT4RS8 16086092 IC50 = 5 nM T65864 CZ2QU1 16086093 IC50 = 277 nM T65864 C13OVU 16086099 IC50 = 50 nM T65864 C2YC0S 16086100 IC50 = 21 nM T65864 C28UZX 16086101 IC50 = 93 nM T65864 CKM8E4 16086102 IC50 = 14 nM T65864 CF0N4J 16086103 IC50 = 139 nM T65864 CKR57M 16086104 IC50 = 9 nM T65864 CI5HJ8 16086105 IC50 = 168 nM T65864 C68SBO 16086106 IC50 = 4 nM T65864 CAYV39 16086107 IC50 = 31 nM T65864 C06NOI 16086108 IC50 = 172 nM T65864 C16NRY 16086114 IC50 = 3 nM T65864 C87TPW 16086115 IC50 = 40 nM T65864 CW35LJ 16086116 IC50 = 25 nM T65864 CA3BD7 16086117 IC50 = 65 nM T65864 C3EKF4 16086118 IC50 = 7 nM T65864 C0QCG4 16086142 IC50 = 57 nM T65864 CCG95S 16099364 IC50 = 38 nM T65864 CE2LR4 16099366 IC50 = 1056 nM T65864 CQG45C 16109001 IC50 = 3700 nM T65864 C1U8XW 16109036 IC50 > 8300 nM T65864 CPS8Y5 16115349 IC50 = 1800 nM T65864 CK1SZ0 16115350 IC50 > 10000 nM T65864 CZL8G5 16115351 IC50 = 450 nM T65864 CRO0D5 16115352 IC50 = 2200 nM T65864 CZ5Y3V 16116847 IC50 = 0.9 nM T65864 CLO43V 16116849 IC50 = 63 nM T65864 C0HO6T 16118191 IC50 = 2 nM T65864 CT92BZ 16118192 IC50 = 4 nM T65864 CIZ6B4 16118193 IC50 = 3 nM T65864 C2CN5O 16118323 IC50 = 22 nM T65864 C4GTU3 16118324 IC50 = 10 nM T65864 CI4E6Y 16118605 IC50 = 6 nM T65864 C8LIW4 16118609 IC50 = 10 nM T65864 CGC34R 16118737 IC50 = 5 nM T65864 CAN2K6 16118739 IC50 = 5 nM T65864 C2Z3XI 16119000 IC50 = 12 nM T65864 CZ08YH 16214904 IC50 > 1600 nM T65864 CNBY51 16415057 IC50 = 4360 nM T65864 CN4X1E 16422038 IC50 > 30000 nM T65864 C0A2JB 16638995 IC50 = 600 nM T65864 CU56EW 16664858 IC50 > 15848.93 nM T65864 C6YK4V 16725338 IC50 = 9 nM T65864 CO5M8A 16726210 IC50 = 0.9 nM T65864 C0H8UN 16730109 Ki = 0.2 nM T65864 CMTS62 16734161 IC50 = 13 nM T65864 CM1C7H 17423309 IC50 = 70 nM T65864 CL9BQ6 17748275 IC50 = 47 nM T65864 CXWY20 17751188 IC50 = 20 nM T65864 C8AH1I 17758019 IC50 = 3600 nM T65864 C1GKL6 17758020 IC50 > 40000 nM T65864 CIE58R 17758239 IC50 > 40000 nM T65864 CO6LR5 17758240 IC50 > 40000 nM T65864 CWH37T 17758574 IC50 > 40000 nM T65864 C57NRL 17759787 IC50 > 40000 nM T65864 C4WMQ2 17892742 IC50 = 3 nM T65864 C43VRU 17898549 IC50 = 173.78 nM T65864 C6AWG3 17898561 IC50 = 85.4 nM T65864 CU35IA 17917696 IC50 = 79 nM T65864 CEQM62 17941443 IC50 = 270 nM T65864 COPZ96 17941451 IC50 = 13 nM T65864 CICQ18 17941464 IC50 = 260 nM T65864 CKE2Y1 17941480 IC50 = 44 nM T65864 CUV3C2 17952492 IC50 > 1000 nM T65864 C4URA6 17981637 IC50 = 7.1 nM T65864 CZIR76 17981640 IC50 = 8.8 nM T65864 CR6A7G 17981652 IC50 = 131 nM T65864 CX6ID5 17981676 IC50 = 6.1 nM T65864 CIQ1W9 17981827 IC50 = 20.4 nM T65864 CX96IH 18322353 IC50 = 44 nM T65864 CCB50Y 18536611 IC50 = 82 nM T65864 C1QUH6 18536613 IC50 = 79 nM T65864 CVGU58 18536615 IC50 = 21.6 nM T65864 CD0UZ5 18536620 IC50 = 119 nM T65864 CZK5O4 18536624 IC50 = 215 nM T65864 CZK08I 18536627 IC50 = 114 nM T65864 CI8Z3Q 18536630 IC50 = 15.14 nM T65864 CY8VG3 18536632 IC50 = 165 nM T65864 C6Y4GF 18536633 IC50 = 40.74 nM T65864 C29GQM 18536638 IC50 = 41 nM T65864 CY06BQ 18536646 IC50 = 10.7 nM T65864 CDS15V 18536647 IC50 = 19 nM T65864 C52SOW 18674213 IC50 = 70.4 nM T65864 C4SPG1 19007057 Ki = 1600 nM T65864 CN6RP1 19013287 IC50 > 30000 nM T65864 CU96LD 19072340 IC50 = 670 nM T65864 C02SWO 19072347 IC50 = 190 nM T65864 CL2K9U 20333093 IC50 > 100000 nM T65864 C6V3PM 20626145 IC50 = 945 nM T65864 C8G5MX 20626557 IC50 = 4.3 nM T65864 C91VRW 20626558 IC50 = 15.3 nM T65864 CDHA15 20626846 IC50 = 25 nM T65864 CN7PI5 20626848 IC50 = 67 nM T65864 CD76FO 20626900 IC50 = 9 nM T65864 C50CPJ 20626915 IC50 = 4 nM T65864 C9H4MK 20626917 IC50 = 40 nM T65864 CSJ08Y 20626953 IC50 = 15 nM T65864 CQJI95 20626977 IC50 = 14 nM T65864 CA92FZ 21027369 IC50 = 170 nM T65864 CSK2J0 21027376 IC50 = 50 nM T65864 CW7I8O 21027446 IC50 = 70 nM T65864 C3D7CB 21078793 Ki = 1500 nM T65864 CR3H9E 21078794 Ki = 1600 nM T65864 CC1E7R 21078798 Ki = 480 nM T65864 C7I9VO 21088983 IC50 = 11 nM T65864 CQB0J9 21088999 IC50 = 60 nM T65864 CIR5V1 21089008 IC50 = 30 nM T65864 CF1A4B 21354185 IC50 = 280 nM T65864 C5UF6X 21354186 IC50 = 160 nM T65864 C06YZB 21354198 IC50 = 970 nM T65864 CVT2Y5 21354200 IC50 = 99 nM T65864 C1RQ6S 21354214 IC50 = 2800 nM T65864 C7OD5R 21354219 IC50 > 20000 nM T65864 C56TNL 21354223 IC50 = 9700 nM T65864 CQ79VS 21354225 IC50 = 260 nM T65864 CRO6A1 21354226 IC50 = 750 nM T65864 CH6BW4 21354227 IC50 = 490 nM T65864 C1Z9BT 21354230 IC50 = 1900 nM T65864 C50BHX 21354231 IC50 = 720 nM T65864 C29PDJ 21354232 IC50 = 210 nM T65864 CFY13E 21354233 IC50 = 200 nM T65864 CI31RU 21354235 IC50 = 3500 nM T65864 CJMN94 21354236 IC50 = 4100 nM T65864 CG29QB 21354237 IC50 = 1000 nM T65864 C3BFQ2 21354238 IC50 > 20000 nM T65864 C6Y0BO 21354245 IC50 = 220 nM T65864 CM79AH 21354254 IC50 = 180 nM T65864 C5BL0G 21867288 IC50 = 508 nM T65864 C2COM8 21867298 IC50 = 2450 nM T65864 CDL0S9 21867310 IC50 = 16 nM T65864 C1B6ZR 21867319 IC50 = 384 nM T65864 CEN6F8 21867330 IC50 = 292 nM T65864 CGE1V7 21867334 IC50 = 68 nM T65864 CHW84A 21867339 IC50 = 48 nM T65864 CB21KJ 21867350 IC50 = 1740 nM T65864 CFCH83 21911291 IC50 = 62 nM T65864 CPN2M4 21911557 IC50 = 39 nM T65864 CM1IF8 21914519 Ki = 9 nM T65864 CK4L1Y 21914620 Ki = 7.943 nM T65864 CZF82E 21914667 Ki = 7.943 nM T65864 CLC7Z6 21922663 IC50 = 420 nM T65864 C6TCO8 21992496 IC50 > 20000 nM T65864 C5EFH7 21992497 IC50 = 59 nM T65864 CO3X7S 21992575 IC50 = 440 nM T65864 COV0S9 21992584 IC50 = 4600 nM T65864 CVD9T3 21992651 IC50 > 20000 nM T65864 C0QS8C 21992678 IC50 = 680 nM T65864 C5N7DG 21992681 IC50 > 20000 nM T65864 CSY41F 21992749 IC50 > 20000 nM T65864 CTF0Q7 21992824 IC50 > 20000 nM T65864 C7KTU1 21992839 IC50 = 9800 nM T65864 C6QNL9 21992913 IC50 = 620 nM T65864 CH73AW 22037206 IC50 = 48.3 nM T65864 CD2H1Z 22037230 IC50 = 68 nM T65864 CXTL58 22037368 IC50 = 71 nM T65864 CC1LM5 22037370 IC50 = 26.5 nM T65864 CK69RD 22037400 IC50 = 39.2 nM T65864 CC7I8U 22037479 IC50 = 25.3 nM T65864 C38GTD 22037512 IC50 = 31.6 nM T65864 CN2XE5 22037660 IC50 = 90 nM T65864 CG4JS7 22037702 IC50 = 70 nM T65864 C1WTP8 22049888 IC50 = 175 nM T65864 CH0C1V 22049899 IC50 = 5 nM T65864 CY56VD 22049940 IC50 = 126 nM T65864 CZ4MA8 22049953 IC50 = 102 nM T65864 CSX50G 22049990 IC50 = 15 nM T65864 C2N1EK 22050003 IC50 = 48.5 nM T65864 C3ZUL4 22050022 IC50 = 55 nM T65864 CI5U1K 22050029 IC50 = 325 nM T65864 CORC80 22050030 IC50 = 3 nM T65864 CG2L3B 22050036 IC50 = 9.5 nM T65864 C9Y8OI 22050098 IC50 = 6 nM T65864 CH1N3O 22050120 IC50 = 12 nM T65864 CL3E5F 22050143 IC50 = 3 nM T65864 CN60BZ 22050201 IC50 = 46 nM T65864 CEYF86 22050254 IC50 = 34 nM T65864 C1M5DE 22050258 IC50 = 6100 nM T65864 C8XSW5 22050265 IC50 = 20 nM T65864 CKI43O 22050310 IC50 = 21 nM T65864 C8H5CM 22050313 IC50 = 8.5 nM T65864 CSY09R 22050346 IC50 = 4 nM T65864 C4MH6A 22050354 IC50 = 251 nM T65864 CI1NV9 22050379 IC50 = 79 nM T65864 CS1OT2 22050381 IC50 = 7 nM T65864 C1WLJ2 22050423 IC50 = 51 nM T65864 CU8L7G 22050426 IC50 = 261 nM T65864 CJ58LI 22050440 IC50 = 250 nM T65864 C13EYW 22050442 IC50 = 50000 nM T65864 CH5FW9 22050449 IC50 = 66 nM T65864 C2YHP0 22050450 IC50 = 8 nM T65864 C09RGX 22050478 IC50 = 49 nM T65864 C2D8XK 22050521 IC50 = 14 nM T65864 CAGM35 22050534 IC50 = 4 nM T65864 C0U3SM 22050546 IC50 = 122 nM T65864 C37XFP 22050621 IC50 = 746 nM T65864 C8ATX9 22050683 IC50 = 8 nM T65864 CM95IS 22050722 IC50 = 59 nM T65864 CSH4R3 22050741 IC50 = 63 nM T65864 C8PX1M 22050760 IC50 = 8 nM T65864 C9WF3I 22050830 IC50 = 3100 nM T65864 C7CK2R 22050837 IC50 = 23 nM T65864 CJ8WU2 22050889 IC50 > 10000 nM T65864 CJO7G4 22051103 IC50 = 17 nM T65864 CUM74N 22051118 IC50 = 72000 nM T65864 CC3OW8 22051155 IC50 = 9 nM T65864 CY6WH0 22051179 IC50 = 681 nM T65864 CJ2YA0 22063896 IC50 = 200 nM T65864 CG3YL1 22063925 IC50 = 9 nM T65864 C3XWK4 22063936 IC50 = 50 nM T65864 CQ2T8N 22066045 IC50 = 152 nM T65864 CFOI16 22129193 IC50 = 170 nM T65864 CO32JV 22238181 IC50 = 416.87 nM T65864 C5IW6G 22242056 IC50 = 9.1 nM T65864 C0UMW7 22262550 IC50 = 82 nM T65864 CR2H9V 22262560 IC50 = 40.5 nM T65864 CKU4L5 22262790 IC50 = 150 nM T65864 CVG5Z0 22291046 IC50 = 30 nM T65864 C8SME4 22291071 IC50 = 310 nM T65864 C4C9WL 22291085 IC50 = 30 nM T65864 CL81JB 22320671 IC50 = 14.6 nM T65864 CF0IQ9 22464113 IC50 = 86 nM T65864 CG6T1C 22464120 IC50 = 83 nM T65864 CU05QJ 22464162 IC50 = 230 nM T65864 CC0AN7 22594077 IC50 = 240 nM T65864 C6KA3X 22594084 IC50 = 210 nM T65864 CJ8GT5 22594093 IC50 = 110 nM T65864 CI5N7X 22631405 IC50 = 3900 nM T65864 C6WE9L 22647873 IC50 = 2 nM T65864 CCSF13 22647899 IC50 = 10.99 nM T65864 CVF0B4 22647905 IC50 = 1.5 nM T65864 CL8J7C 22647927 IC50 = 6 nM T65864 CWOM34 22647945 IC50 = 0.7 nM T65864 CRTE24 22648022 IC50 = 0.1 nM T65864 COBY76 22648115 IC50 = 1.4 nM T65864 C4WG0Q 22648138 IC50 = 1 nM T65864 C4ONH2 22648169 IC50 = 5.998 nM T65864 CA82VX 22648176 IC50 = 3 nM T65864 C0RZE7 22648190 IC50 = 0.5 nM T65864 CC1U4X 22732253 IC50 = 140 nM T65864 C1KYD0 22732319 IC50 = 510 nM T65864 CN76KY 22953580 IC50 = 80 nM T65864 CIVA91 22953801 IC50 = 70 nM T65864 C5NJD7 22953832 IC50 = 54.7 nM T65864 C8EJ1X 22987996 IC50 = 3 nM T65864 C9BI2Y 23060924 IC50 > 1100 nM T65864 C2NLE3 23060985 IC50 > 1100 nM T65864 CG1I9K 23133388 IC50 = 9.6 nM T65864 C34QYK 23400138 IC50 = 5 nM T65864 C8TI7M 23400141 IC50 = 3 nM T65864 CR9L5X 23400156 IC50 = 11 nM T65864 C27UJN 23400158 IC50 = 6 nM T65864 CHV2K1 23400159 IC50 = 9 nM T65864 CBR20T 23400164 IC50 = 9 nM T65864 CD3A8N 23400169 IC50 = 13 nM T65864 C2JBU8 23400177 IC50 = 7 nM T65864 CZ9V8T 23400179 IC50 = 3 nM T65864 CBK34Y 23400206 IC50 = 8 nM T65864 CM50DA 23400207 IC50 = 18 nM T65864 C75DWA 23400208 IC50 = 14 nM T65864 CY1QB9 23400210 IC50 = 24 nM T65864 CS36ND 23400211 IC50 = 67 nM T65864 CPXG60 23400213 IC50 = 253 nM T65864 C8KJO4 23400214 IC50 = 10 nM T65864 C2DX7W 23400215 IC50 = 6 nM T65864 C7D9LI 23400216 IC50 = 4 nM T65864 C54NCG 23400217 IC50 = 12 nM T65864 CSP35V 23400218 IC50 = 13 nM T65864 C79GOA 23400222 IC50 = 184 nM T65864 C8LFY6 23400224 IC50 = 21 nM T65864 CJRL54 23400251 IC50 = 4 nM T65864 C2LWT7 23433710 IC50 = 83.2 nM T65864 C0B8JU 23433737 IC50 = 22.3 nM T65864 CMU2T8 23433741 IC50 = 17.7 nM T65864 CI7F1U 23433744 IC50 = 37.8 nM T65864 CPB13I 23433758 IC50 = 4.6 nM T65864 CNCB29 23433767 IC50 = 544 nM T65864 C06EWU 23433778 IC50 = 13.5 nM T65864 COHK54 23433783 IC50 = 12.4 nM T65864 CFT4H3 23434538 IC50 = 1 nM T65864 CSKH65 23434573 IC50 = 594 nM T65864 C7IVP6 23434577 IC50 = 106 nM T65864 CG1P2J 23434580 IC50 = 15 nM T65864 CTV6K2 23434654 IC50 = 42 nM T65864 CH49JD 23443327 IC50 = 180 nM T65864 C57AHM 23443377 IC50 = 180 nM T65864 C6K8HD 23532566 IC50 = 0.77 nM T65864 CE7K3W 23532567 IC50 = 0.2 nM T65864 C9VBX2 23532568 IC50 = 0.5998 nM T65864 CWFC29 23532607 IC50 = 0.84 nM T65864 CELR52 23532663 IC50 = 1.199 nM T65864 C4X1WC 23532664 IC50 = 0.6 nM T65864 C5KY6F 23532666 IC50 = 0.5 nM T65864 C1C8EF 23532667 IC50 = 0.38 nM T65864 C1K6TP 23532674 IC50 = 2.4 nM T65864 C5UD9Z 23532675 IC50 = 0.27 nM T65864 CND3A5 23532688 IC50 = 0.51 nM T65864 CC5YA9 23532689 IC50 = 0.61 nM T65864 CH4W9B 23532696 IC50 = 1 nM T65864 C7AE8G 23532702 IC50 = 0.5 nM T65864 CR3GI1 23532736 IC50 = 1.8 nM T65864 CJ1GE9 23532737 IC50 = 6.4 nM T65864 CM5L3K 23532793 IC50 = 0.9 nM T65864 CDE6J9 23532851 IC50 = 0.45 nM T65864 CV50CQ 23532872 IC50 = 2.59 nM T65864 CAK9J8 23532873 IC50 = 28 nM T65864 C5AZ7B 23536770 IC50 = 463 nM T65864 CR7DC6 23546124 IC50 = 7900 nM T65864 C3XFN0 23551786 IC50 = 21 nM T65864 CL14EK 23581364 IC50 = 30 nM T65864 CWG94O 23581368 IC50 = 1250 nM T65864 C3TRK1 23581376 IC50 = 200 nM T65864 CJ85GZ 23581379 IC50 = 800 nM T65864 C78GIA 23581385 IC50 = 100 nM T65864 CWLD49 23581392 IC50 = 70 nM T65864 CNMY82 23581397 IC50 = 140 nM T65864 CW97ZG 23581402 IC50 = 15800 nM T65864 C5HEG6 23581403 IC50 = 1500 nM T65864 CJ9AH3 23581414 IC50 = 200 nM T65864 CK4F1R 23581416 IC50 = 140 nM T65864 CBM5U6 23581418 IC50 = 70 nM T65864 C8MP1T 23581427 IC50 = 6200 nM T65864 C3BY2D 23581428 IC50 = 290 nM T65864 CX15YT 23581429 IC50 = 260 nM T65864 C8VN2P 23581434 IC50 = 1800 nM T65864 CYB92N 23581647 IC50 = 540 nM T65864 C90IFU 23581649 IC50 = 370 nM T65864 C4IDA7 23581655 IC50 = 380 nM T65864 CM6B7E 23581658 IC50 = 500 nM T65864 C98HSM 23581659 IC50 = 390 nM T65864 CYV59W 23581662 IC50 > 32000 nM T65864 CB92DO 23581664 IC50 = 680 nM T65864 CXF1Y8 23581665 IC50 = 8000 nM T65864 CRB0A7 23581668 IC50 = 140 nM T65864 C18NMX 23581670 IC50 = 270 nM T65864 CR3M1N 23644582 Ki = 400 nM T65864 CWT7R6 23644699 IC50 = 25 nM T65864 COT5Q4 23647065 IC50 > 1000 nM T65864 CQ28DG 23647066 IC50 = 100 nM T65864 C41VBR 23647067 IC50 = 4000 nM T65864 C68WQX 23647068 IC50 = 60 nM T65864 C9D8ZL 23647069 IC50 = 2500 nM T65864 C20RXS 23647070 IC50 = 680 nM T65864 CE4D6B 23647071 IC50 = 12500 nM T65864 CW19FP 23647072 IC50 > 1000 nM T65864 CX75TK 23647073 IC50 > 1000 nM T65864 C6TJ1P 23647074 IC50 = 14400 nM T65864 C70PNO 23647075 IC50 = 690 nM T65864 C6A9UT 23647076 IC50 > 1000 nM T65864 CMTC30 23647077 IC50 = 260 nM T65864 C5PQ8U 23647078 IC50 = 90 nM T65864 C7SQ8C 23647316 IC50 = 3 nM T65864 CKV70B 23647317 IC50 = 2.2 nM T65864 C0YCE4 23647318 IC50 = 5.1 nM T65864 CG6D4M 23647319 IC50 = 2.5 nM T65864 C1QIN6 23647320 IC50 = 43.2 nM T65864 CR2F7K 23647321 IC50 = 26.4 nM T65864 CB56TE 23647322 IC50 = 8.3 nM T65864 CGDW05 23647323 IC50 = 14.5 nM T65864 CXN8E7 23647324 IC50 = 24.5 nM T65864 CRW25S 23647325 IC50 = 5.6 nM T65864 C46TSL 23647326 IC50 = 8 nM T65864 CVEF76 23647327 IC50 = 5.4 nM T65864 C0GN9E 23647328 IC50 = 9.2 nM T65864 CM6IG0 23647329 IC50 = 19.5 nM T65864 CY8Z7X 23647330 IC50 = 7.6 nM T65864 CWI0Y1 23647331 IC50 = 55.5 nM T65864 C54JRP 23647332 IC50 = 8.8 nM T65864 C4KC1J 23647333 IC50 = 5.5 nM T65864 CD2V5Z 23647334 IC50 = 198 nM T65864 CZ5M9O 23647335 IC50 = 4.7 nM T65864 CN18GD 23647336 IC50 = 17.9 nM T65864 CP63DB 23647337 IC50 = 14 nM T65864 C5BO6N 23647338 IC50 = 15.4 nM T65864 CTRK81 23647339 IC50 = 0.4 nM T65864 C43ZVU 23647340 IC50 = 0.4 nM T65864 CL5B6O 23647341 IC50 = 3.5 nM T65864 CW5C7Q 23647342 IC50 = 11.8 nM T65864 CQ14ZE 23647343 IC50 = 19.9 nM T65864 CPQ2C3 23647344 IC50 = 3.75 nM T65864 C49KWO 23647345 IC50 = 1.1 nM T65864 CVS15P 23647346 IC50 = 1.5 nM T65864 CA8V9B 23647347 IC50 = 2.5 nM T65864 C4XD8H 23647348 IC50 = 2.8 nM T65864 CNV8S5 23647349 IC50 = 33.2 nM T65864 C2T1LI 23647350 IC50 = 6.2 nM T65864 C7TSR0 23647364 IC50 = 790 nM T65864 CHI73F 23647365 IC50 = 560 nM T65864 CY34HX 23647366 IC50 = 760 nM T65864 C7Z0LW 23647367 IC50 = 2400 nM T65864 C8S9KH 23647368 IC50 = 140 nM T65864 COEA71 23647369 IC50 = 310 nM T65864 C3QI0B 23647370 IC50 = 2000 nM T65864 CQ14UH 23647371 IC50 = 3500 nM T65864 CLW83Z 23647372 IC50 = 168 nM T65864 C0PN6O 23647373 IC50 = 197 nM T65864 C0U7GT 23647374 IC50 = 490 nM T65864 C4EX0K 23647375 IC50 = 20 nM T65864 C9G0TU 23647376 IC50 = 35 nM T65864 CQP59Z 23647378 IC50 = 8 nM T65864 C5KEF4 23647379 IC50 = 20 nM T65864 CWH9Z2 23647628 IC50 = 0.2 nM T65864 CQ39NA 23647629 IC50 = 10 nM T65864 CE2FJ3 23647630 IC50 = 4.2 nM T65864 C2KQL8 23647631 IC50 = 5.3 nM T65864 C6B2FV 23647632 IC50 = 2 nM T65864 CA7G3K 23647633 IC50 = 3 nM T65864 C6XNF7 23647634 IC50 = 1.1 nM T65864 CI93JV 23647635 IC50 = 0.8 nM T65864 CZX86H 23647636 IC50 = 1.9 nM T65864 C7FL3O 23647637 IC50 = 4 nM T65864 CPA7M5 23647638 IC50 = 2 nM T65864 CH27WV 23647639 IC50 = 5.6 nM T65864 CNM0T6 23647640 IC50 = 4.2 nM T65864 CK2B5V 23647641 IC50 = 0.5 nM T65864 CF58LA 23647642 IC50 = 1 nM T65864 CA84MR 23647643 IC50 = 20 nM T65864 C9UE6H 23647644 IC50 = 4 nM T65864 CQ0GU6 23647645 IC50 = 2 nM T65864 C7Q9TJ 23647646 IC50 = 2 nM T65864 CB41HK 23647647 IC50 = 1.2 nM T65864 CV1FS4 23647648 IC50 = 0.5 nM T65864 CN9H8P 23647649 IC50 = 0.7 nM T65864 CDMI50 23661564 IC50 > 100000 nM T65864 CBGC24 23729163 IC50 <= 2 nM T65864 CBP1W2 24180462 IC50 = 11 nM T65864 CN9S3A 24517908 IC50 = 2100 nM T65864 CNYO87 24744181 IC50 = 5 nM T65864 CH1L5D 24744497 IC50 = 24 nM T65864 C1E7QT 24744663 IC50 = 24 nM T65864 C39KYC 24745286 IC50 = 17 nM T65864 CPR70N 24745453 IC50 = 2530 nM T65864 CT64ZV 24745605 IC50 = 23 nM T65864 CV9U8E 24745781 IC50 = 21 nM T65864 CA9N8F 24745785 IC50 = 208 nM T65864 C6SV4Y 24745787 IC50 = 39 nM T65864 CH80BE 24745950 IC50 = 228 nM T65864 CIF4M5 24745952 IC50 = 802 nM T65864 CL49UD 24745955 IC50 = 17 nM T65864 C72LGH 24746115 IC50 = 37 nM T65864 C8J3FZ 24746297 IC50 = 126 nM T65864 CAG7M1 24746299 IC50 = 38 nM T65864 C4YFK7 24746456 IC50 = 14 nM T65864 CX09TL 24746457 IC50 = 20 nM T65864 CN94TV 24746459 IC50 = 491 nM T65864 C23ODH 24746612 IC50 = 42 nM T65864 C96QEC 24746614 IC50 = 70 nM T65864 CVW08C 24754377 IC50 = 4.7 nM T65864 C1LR6W 24754378 IC50 = 7.7 nM T65864 CE45LK 24754379 IC50 = 5.6 nM T65864 C4D6YQ 24755185 IC50 = 220 nM T65864 CMQ5A4 24755186 IC50 = 1.1 nM T65864 C7RN3M 24755187 IC50 = 78 nM T65864 CADH96 24755189 IC50 = 4 nM T65864 C6VQ2I 24755247 IC50 = 42 nM T65864 C1GY9S 24755250 IC50 = 23 nM T65864 CIO7G9 24755251 IC50 = 3.3 nM T65864 CEGM85 24755252 IC50 = 1.5 nM T65864 CCY8E2 24755328 IC50 = 1.2 nM T65864 CN6L0Y 24755331 IC50 = 3.6 nM T65864 CM3K8R 24755332 IC50 = 13 nM T65864 C2CL5R 24755333 IC50 = 13 nM T65864 C04WKM 24755388 IC50 = 12 nM T65864 CV15ZO 24755390 IC50 = 15 nM T65864 CYL2R9 24755391 IC50 = 5.5 nM T65864 CB2H3V 24755452 IC50 = 680 nM T65864 C9OEN0 24755454 IC50 = 20 nM T65864 CZG15T 24755455 IC50 = 230 nM T65864 CD0M3C 24755476 IC50 = 6.4 nM T65864 C7YG1N 24759534 IC50 = 1200 nM T65864 CT56IM 24764438 Ki = 0.46 nM T65864 CQNP54 24764449 IC50 = 100000 nM T65864 C2UOE0 24766030 IC50 > 50000 nM T65864 C6UVG5 24772976 IC50 = 3 nM T65864 CSFN69 24788015 IC50 = 4050 nM T65864 C2IA1Y 24794468 IC50 = 2 nM T65864 C64KZL 24797480 IC50 = 6.5 nM T65864 CW9E5O 24797670 IC50 = 1 nM T65864 CLBP72 24798571 IC50 > 10000 nM T65864 CI2ZH0 24805930 IC50 = 11 nM T65864 CBH9L2 24805931 IC50 = 18 nM T65864 C54LVP 24805932 IC50 = 6 nM T65864 CW89YV 24806129 IC50 = 37 nM T65864 CLR8E6 24806130 IC50 = 2 nM T65864 CIWK42 24807346 IC50 = 41 nM T65864 CW9NZ1 24807347 IC50 = 87 nM T65864 C0Y5HS 24807348 IC50 = 27 nM T65864 CA78WR 24807349 IC50 = 13 nM T65864 CL2YR8 24807350 IC50 = 15 nM T65864 CLG3Z4 24807351 IC50 = 5 nM T65864 CKVN06 24807540 IC50 = 3 nM T65864 CY53ZJ 24807541 IC50 = 12 nM T65864 CEM36Q 24807542 IC50 = 10 nM T65864 CHM90F 24807544 IC50 = 3 nM T65864 CU9CG5 24807724 IC50 = 3 nM T65864 COP0B4 24810673 IC50 = 11 nM T65864 C16DKC 24810995 IC50 > 3000 nM T65864 CC8Y1U 24810996 IC50 > 3000 nM T65864 CH21WG 24810997 IC50 = 2100 nM T65864 CQ1D8M 24810999 IC50 = 9300 nM T65864 CNI4W8 24811099 IC50 > 30000 nM T65864 C0MXK3 24811100 IC50 = 2600 nM T65864 CFZN51 24811101 IC50 = 1200 nM T65864 CRF71M 24811102 IC50 = 1500 nM T65864 CB8A2T 24811103 IC50 > 30000 nM T65864 CP6N9M 24812718 IC50 = 998 nM T65864 CM72QB 24821653 IC50 = 0.95 nM T65864 C2G7PB 24821851 IC50 = 84 nM T65864 CQY2V9 24821915 IC50 = 24 nM T65864 CY3QC9 24821916 IC50 = 31 nM T65864 CBEM80 24821917 IC50 = 64 nM T65864 CWZK03 24821918 IC50 = 8 nM T65864 C73QOF 24821919 IC50 = 16 nM T65864 C3BJ2V 24821979 IC50 = 51 nM T65864 CCP2M3 24822704 IC50 > 50000 nM T65864 CYBI02 24823426 IC50 = 87 nM T65864 C45UGH 24823586 IC50 = 10 nM T65864 CFA3T8 24823588 IC50 = 179 nM T65864 C51ZTV 24823589 IC50 = 8 nM T65864 CX0QC1 24823590 IC50 = 12 nM T65864 CR7CH6 24823736 IC50 = 1070 nM T65864 C26KXV 24823738 IC50 = 103 nM T65864 CO3K7R 24823740 IC50 = 6 nM T65864 CBLJ48 24823898 IC50 = 233 nM T65864 CG0K1Z 24824046 IC50 = 200 nM T65864 C2LPM3 24829378 IC50 = 480 nM T65864 CRPO60 24853743 IC50 = 3830 nM T65864 C6C4WV 24853802 IC50 = 3900 nM T65864 CNX48L 24853803 IC50 = 1150 nM T65864 CKJQ40 24853806 IC50 = 230 nM T65864 CRJ1S9 24853807 IC50 = 350 nM T65864 C48AFX 24853808 IC50 = 970 nM T65864 C8QF0V 24853871 IC50 = 1400 nM T65864 CB2Y1J 24853876 IC50 = 1630 nM T65864 CK4CG5 24853877 IC50 = 2130 nM T65864 C0V3GD 24853956 IC50 = 1320 nM T65864 CGN0U9 24853957 IC50 = 2500 nM T65864 C4E7TP 24853959 IC50 = 320 nM T65864 CX0S9L 24854902 IC50 = 0.8 nM T65864 C1SVT2 24854903 IC50 = 1 nM T65864 C61KPI 24856363 Ki = 9 nM T65864 CH1YI6 24856364 Ki = 4.4 nM T65864 CCS58O 24863072 IC50 = 110 nM T65864 C6C2GX 24863500 IC50 = 350 nM T65864 CYVB83 24863584 IC50 = 450 nM T65864 CQ15ML 24863670 IC50 = 51 nM T65864 C4XZ3N 24863671 IC50 > 1600 nM T65864 C4MG3B 24882476 IC50 = 856 nM T65864 C13QYB 24884503 IC50 = 216 nM T65864 CRG15B 24893986 IC50 = 27.6 nM T65864 CW0MT7 24893987 IC50 = 101 nM T65864 C4S7CP 24893988 IC50 = 31 nM T65864 C5A6PI 24894128 IC50 = 3 nM T65864 CO7YQ6 24896765 IC50 = 141 nM T65864 CY8L7E 24896769 IC50 = 14 nM T65864 C5XS7N 24897233 IC50 = 0.72 nM T65864 CE3HW0 24897234 IC50 = 0.59 nM T65864 CD0L1Z 24897447 IC50 = 0.49 nM T65864 CT3HF9 24897657 IC50 = 0.53 nM T65864 C8S3CZ 24897658 IC50 = 0.27 nM T65864 CXCM54 24897876 IC50 = 77 nM T65864 CDPU54 24898309 IC50 > 10000 nM T65864 CF5X3J 24898310 IC50 > 10000 nM T65864 CE13YZ 24898751 IC50 = 0.28 nM T65864 CR49LI 24899731 IC50 = 148 nM T65864 CQ69KH 24899732 IC50 = 66 nM T65864 C6IG5T 24899733 IC50 = 68 nM T65864 CH61IV 24899735 IC50 = 144 nM T65864 C4K6BX 24899987 IC50 = 0.82 nM T65864 C8H3FA 24900230 IC50 = 41 nM T65864 C9OSB6 24900231 IC50 = 333 nM T65864 CPLA45 24900232 IC50 = 195 nM T65864 C5Y6GM 24901423 IC50 = 300 nM T65864 C8RUK7 24905709 IC50 = 47 nM T65864 C8DG6O 24905757 IC50 = 13 nM T65864 C7DY8U 24905758 IC50 = 2150 nM T65864 C4UHZ6 24905759 IC50 = 82 nM T65864 C12TCX 24905760 IC50 = 282 nM T65864 CJM94C 24905761 IC50 = 248 nM T65864 C97YFX 24905762 IC50 = 46 nM T65864 CZ1VP4 24905809 IC50 = 314 nM T65864 CRBD03 24905810 IC50 = 113 nM T65864 CZI65E 24905811 IC50 = 119 nM T65864 CU03RT 24905812 IC50 = 191 nM T65864 C5S2PI 24905813 IC50 = 153 nM T65864 CD5L3J 24905814 IC50 = 15 nM T65864 CZI9N1 24905857 IC50 = 23 nM T65864 CUP7O2 24905858 IC50 = 126 nM T65864 CV1D7F 24905859 IC50 = 26 nM T65864 C7YRW2 24905860 IC50 = 36 nM T65864 CC3J9T 24905861 IC50 = 45 nM T65864 CLGP50 24905862 IC50 = 6 nM T65864 COA42F 24905863 IC50 = 34 nM T65864 CWP0M9 24905905 IC50 = 61 nM T65864 C45YBP 24905906 IC50 = 639 nM T65864 C7QVK2 24905907 IC50 = 542 nM T65864 CG4EW9 24905908 IC50 = 641 nM T65864 C5PNC0 24905909 IC50 = 292 nM T65864 CBIQ08 24905910 IC50 = 68 nM T65864 C7C5EV 24905956 IC50 = 28 nM T65864 CA3L8X 24905957 IC50 = 17 nM T65864 CK4SL6 24905958 IC50 = 348 nM T65864 C7IEC3 24905959 IC50 = 1340 nM T65864 CC24VE 24905960 IC50 = 173 nM T65864 CZ6K8S 24905961 IC50 = 171 nM T65864 CBT42M 24906013 IC50 = 199 nM T65864 C83RWS 24906014 IC50 = 93 nM T65864 CL31XQ 24906015 IC50 = 49 nM T65864 C8RSF0 24906016 IC50 = 23 nM T65864 CZE4N6 24906017 IC50 = 60 nM T65864 CSH5J2 24906018 IC50 = 70 nM T65864 CMT14N 24906062 IC50 = 98 nM T65864 C46EXD 24906063 IC50 = 239 nM T65864 CJD73S 24906064 IC50 = 80 nM T65864 CW1FE0 24906065 IC50 = 27 nM T65864 COI13A 24906066 IC50 = 13 nM T65864 CL5J7O 24906107 IC50 = 90 nM T65864 CF09XG 24906108 IC50 = 11 nM T65864 CHFV23 24906109 IC50 = 230 nM T65864 CT4WS5 24906110 IC50 = 20 nM T65864 CAF0M5 24906111 IC50 = 34 nM T65864 C06EKN 24906112 IC50 = 21 nM T65864 CO97UZ 24906113 IC50 = 35 nM T65864 CQG8T9 24906150 IC50 = 10 nM T65864 C93KCS 24906151 IC50 = 15 nM T65864 CI82OW 24906152 IC50 = 436 nM T65864 CF19ZB 24906153 IC50 = 33 nM T65864 C2OI3T 24906154 IC50 = 87 nM T65864 C8DG1Y 24941253 Ki = 0.4 nM T65864 C6CVK4 24959046 IC50 > 100000 nM T65864 CU7I2E 24963046 IC50 = 0.9 nM T65864 C2FEL5 24965752 IC50 = 33 nM T65864 CB5VC1 24966097 IC50 = 42 nM T65864 CEM91Y 24966100 IC50 = 28 nM T65864 C5PV9L 24967901 IC50 = 51 nM T65864 CFY08G 24968590 IC50 = 22 nM T65864 C9BGM8 24968591 IC50 = 60 nM T65864 CMJ3H5 24968592 IC50 = 78 nM T65864 CGE5U3 24968594 IC50 = 190 nM T65864 C9U8QN 24968751 IC50 = 56 nM T65864 C4CWQ9 24985573 IC50 = 4.8 nM T65864 CA01UI 24985915 IC50 = 0.2 nM T65864 C4EG8R 24993189 IC50 > 10000 nM T65864 C1BZO9 25005874 IC50 = 10.8 nM T65864 CL7G3C 25009302 IC50 = 9 nM T65864 CNR41J 25016226 IC50 = 0.9 nM T65864 CI7ZE2 25023830 IC50 = 3740 nM T65864 CBYX96 25030803 IC50 = 29 nM T65864 CVQS96 25052767 Ki = 1.4 nM T65864 CSI0K4 25059579 IC50 = 2.5 nM T65864 CDPX75 25093461 Ki = 490 nM T65864 CI6MF0 25093462 Ki = 250 nM T65864 C7MG0P 25093463 Ki = 100 nM T65864 C4E1XB 25093464 Ki = 40 nM T65864 C7TS0Z 25093465 Ki = 100 nM T65864 C9LV1E 25093466 Ki = 140 nM T65864 C0CSV1 25093467 Ki > 2500 nM T65864 C3GT0P 25093468 Ki = 1600 nM T65864 C47FHP 25093469 Ki > 2500 nM T65864 C7Q2RV 25093470 Ki > 2500 nM T65864 C1PE8Z 25093471 Ki = 2000 nM T65864 CL40XH 25093472 Ki = 1700 nM T65864 C9TB6U 25093473 Ki = 220 nM T65864 CF64LW 25093474 Ki > 2500 nM T65864 CSA6V4 25093475 Ki > 2500 nM T65864 CKR0Y5 25107839 IC50 = 215 nM T65864 CB0XU8 25107840 IC50 = 184 nM T65864 CS87CF 25107841 IC50 = 487 nM T65864 CT0AQ6 25107842 IC50 = 158 nM T65864 CU1R8T 25107843 IC50 = 1220 nM T65864 CB1OI3 25107844 IC50 = 102 nM T65864 C60VRS 25107845 IC50 = 2 nM T65864 CVO97P 25113874 IC50 = 33 nM T65864 C3NJS0 25113875 IC50 = 29 nM T65864 CQG39V 25114098 IC50 = 37 nM T65864 CLXC40 25116627 IC50 = 2.7 nM T65864 CN8P9B 25118219 Ki = 1.9 nM T65864 CD8B9A 25118220 Ki = 2.3 nM T65864 C2MOG6 25118568 Ki = 0.9 nM T65864 C3HB6S 25118571 Ki = 0.8 nM T65864 CV4Y6Z 25118573 Ki = 1 nM T65864 CY14DU 25119291 Ki = 1.1 nM T65864 C0K1OR 25119294 Ki = 1.9 nM T65864 CC14NJ 25119643 Ki = 1.7 nM T65864 CQGP36 25119645 Ki = 1.5 nM T65864 CG8D5U 25119991 Ki = 0.6 nM T65864 CTV54O 25123227 IC50 > 10000 nM T65864 CG9LW7 25123829 IC50 = 130 nM T65864 CG3XC9 25124150 IC50 = 440 nM T65864 CQ2I9A 25124305 IC50 = 950 nM T65864 CIJM32 25124640 Ki = 90 nM T65864 CO2IR5 25124816 IC50 = 11000 nM T65864 C1IYN7 25127854 IC50 > 1000 nM T65864 CKD14B 25127856 IC50 > 1000 nM T65864 CJBX60 25128180 IC50 > 1000 nM T65864 CC5SD9 25128181 IC50 > 1000 nM T65864 CF7C5B 25129829 IC50 = 1.9 nM T65864 CXNM84 25129830 IC50 = 1.2 nM T65864 CY2S1P 25129831 IC50 = 182 nM T65864 C1NPM8 25130181 IC50 = 0.6 nM T65864 CD29CQ 25133018 IC50 = 1107 nM T65864 CQMU82 25138148 IC50 = 1 nM T65864 CD9O6K 25138149 IC50 = 28 nM T65864 CM6XF2 25138294 EC50 = 14800 nM T65864 CTO24B 25174101 IC50 = 170 nM T65864 CEA5R6 25181471 IC50 = 100000 nM T65864 CL0Z1F 25181502 Ki = 0.4 nM T65864 CB4CI5 25194890 Ki = 2 nM T65864 CA9T7Y 25195321 EC50 = 46300 nM T65864 C5PC2Z 25195322 EC50 = 57800 nM T65864 CW1A4N 25196726 IC50 > 100000 nM T65864 CPY2C9 25203945 IC50 = 12589.25 nM T65864 CLFM35 25206064 IC50 > 50000 nM T65864 C6FGQ1 25206346 IC50 = 45 nM T65864 C41MJN 25210518 IC50 = 1100 nM T65864 CC6HK7 25210519 IC50 = 150 nM T65864 CFU8G9 25210521 IC50 = 120 nM T65864 CNG96H 25210579 IC50 > 10000 nM T65864 C1UMI4 25242389 IC50 = 3.3 nM T65864 CC7GX8 25253556 IC50 = 2700 nM T65864 C56XDP 25257469 IC50 = 1080 nM T65864 C8SOW7 25257470 IC50 = 310 nM T65864 CTP92K 25257471 IC50 = 240 nM T65864 CYE46B 25257472 IC50 = 440 nM T65864 CB82GX 25257706 IC50 = 2730 nM T65864 CS98QU 25257707 IC50 = 180 nM T65864 CEK14U 25257708 IC50 = 1950 nM T65864 CT7I0D 25257709 IC50 = 330 nM T65864 C0JAI5 25257710 IC50 = 1190 nM T65864 C5SNQ8 25257711 IC50 = 2680 nM T65864 CGQ8D3 25270849 IC50 = 1 nM T65864 CES46M 25270850 IC50 = 1.1 nM T65864 CN7S0V 25271185 IC50 = 4 nM T65864 CE3T0R 25271186 IC50 = 2.9 nM T65864 CE0PX2 42601396 IC50 = 800 nM T65864 C2IOM6 42605758 IC50 = 273 nM T65864 CC28KA 42606570 IC50 = 1.2 nM T65864 CGV34B 42608443 IC50 = 370 nM T65864 CM0C2R 42608444 IC50 = 320 nM T65864 C2FU9P 42618077 IC50 > 100000 nM T65864 CWS37O 42618140 IC50 > 25118.86 nM T65864 C2JV3O 42618143 IC50 > 25118.86 nM T65864 CG01BO 42618144 IC50 > 25118.86 nM T65864 CU9E4P 42629114 IC50 > 10000 nM T65864 CL26DF 42640797 IC50 <= 2 nM T65864 C8M6NY 42640798 IC50 = 15 nM T65864 CNK78M 42640802 EC50 = 2700 nM T65864 CIOR58 42640803 EC50 <= 8 nM T65864 CA7I0F 42647297 IC50 = 3.2 nM T65864 CCB1E9 44124695 IC50 = 6 nM T65864 CO42DC 44138048 IC50 = 7943.28 nM T65864 CL65QV 44138049 IC50 = 7943.28 nM T65864 CWXJ06 44156975 IC50 > 100000 nM T65864 C58KSV 44156976 IC50 > 100000 nM T65864 CLW80F 44160269 IC50 = 32000 nM T65864 CDW4F2 44186373 IC50 = 1800 nM T65864 CWT68J 44186427 IC50 = 1000 nM T65864 CCFQ29 44187005 IC50 = 145 nM T65864 C8KNA3 44219632 Ki > 4000 nM T65864 C0VIX4 44219633 Ki > 4000 nM T65864 CK73NR 44219749 IC50 > 50000 nM T65864 CEL61X 44229839 IC50 > 10000 nM T65864 C2WH0M 44249910 IC50 = 967 nM T65864 CU7TQ4 44249911 IC50 = 411 nM T65864 C0SPV1 44250043 IC50 = 174 nM T65864 C4CF6Z 44250044 IC50 = 149 nM T65864 CBD82X 44250045 IC50 = 1655 nM T65864 CC45SQ 44250046 IC50 = 15 nM T65864 C2CT7Q 44250342 IC50 = 0.9 nM T65864 CJ75IB 44250343 IC50 = 1.65 nM T65864 C42MJN 44250344 IC50 = 0.09 nM T65864 C79TPC 44250345 IC50 = 4570 nM T65864 CTUL86 44250346 IC50 = 0.08 nM T65864 C7F4QU 44250416 IC50 = 75 nM T65864 CJ28CO 44250418 IC50 = 5.2 nM T65864 C7NYB5 44250420 IC50 = 1 nM T65864 C4H8FS 44250482 IC50 = 1.8 nM T65864 C8HSF0 44250483 IC50 = 0.9 nM T65864 CVFT50 44250484 IC50 = 1.4 nM T65864 CJRU72 44250547 IC50 = 128 nM T65864 C7F6HZ 44250548 IC50 = 8 nM T65864 CQP27S 44250549 IC50 = 544 nM T65864 CS2CK9 44250550 IC50 = 1.8 nM T65864 COV52B 44250616 IC50 = 86 nM T65864 C5EUT4 44250618 IC50 = 2.3 nM T65864 C9L0AN 44250620 IC50 = 0.8 nM T65864 C18QZL 44250621 IC50 = 72 nM T65864 CL63JW 44250622 IC50 = 7.4 nM T65864 CG60EM 44250685 IC50 = 18 nM T65864 CO37WN 44250686 IC50 = 9 nM T65864 C2MQ7P 44250687 IC50 = 135 nM T65864 CM5GN3 44250753 IC50 = 2 nM T65864 CVTJ05 44250757 IC50 = 4.7 nM T65864 CH1V4Q 44250817 IC50 = 32 nM T65864 CPI7Y2 44250878 IC50 = 583 nM T65864 C65OKN 44250879 IC50 = 741 nM T65864 CC39DR 44250880 IC50 = 880 nM T65864 C8YV7W 44250881 IC50 = 173 nM T65864 CLY1A3 44251218 IC50 = 1.3 nM T65864 CY4JW3 44251219 IC50 = 130 nM T65864 C3X6BQ 44251220 IC50 = 1.4 nM T65864 CZ62FW 44251221 IC50 = 20 nM T65864 CBU07V 44251292 IC50 = 12 nM T65864 CX91IA 44251293 IC50 = 9 nM T65864 CL7X1U 44251295 IC50 = 10 nM T65864 C0WCE2 44251296 IC50 = 3 nM T65864 CYI5T1 44251297 IC50 = 275 nM T65864 CLY78F 44251298 IC50 = 6 nM T65864 CCM6A4 44251365 IC50 = 0.22 nM T65864 C9JAK6 44251366 IC50 = 1166 nM T65864 CF3W6Y 44251367 IC50 = 2 nM T65864 CM0T3L 44251368 IC50 = 1.2 nM T65864 C4L7DH 44251369 IC50 = 150 nM T65864 CJG90M 44251370 IC50 = 5 nM T65864 C7TH6G 44251598 IC50 = 0.06 nM T65864 C0C7VH 44269190 IC50 = 602.56 nM T65864 CZ1IC4 44269212 IC50 = 312 nM T65864 C1C3QM 44269241 IC50 = 209 nM T65864 C6SUK7 44269247 IC50 = 220 nM T65864 CQF3R0 44269251 IC50 = 453 nM T65864 C2D8QF 44269252 IC50 = 406 nM T65864 C9OHA5 44269265 IC50 = 300 nM T65864 C1SH4K 44269269 IC50 = 189 nM T65864 CMG14K 44269272 IC50 = 75 nM T65864 C72UPN 44269291 IC50 = 151 nM T65864 CR4JD5 44271834 IC50 = 82 nM T65864 CY83FE 44271855 IC50 = 16 nM T65864 C3E1OW 44271856 IC50 = 550 nM T65864 C2A6EW 44271857 IC50 = 30 nM T65864 CN7SB3 44271872 IC50 = 510 nM T65864 CAKX19 44272022 IC50 > 16700 nM T65864 CIV34W 44272034 IC50 = 140 nM T65864 C6OM5W 44272036 IC50 = 56 nM T65864 CFO97Z 44272038 IC50 = 180 nM T65864 CQS82P 44272046 IC50 = 2100 nM T65864 CK8LS9 44272047 IC50 = 350 nM T65864 CTB28G 44272048 IC50 = 57 nM T65864 C5TJL2 44272053 IC50 = 26 nM T65864 CD7LW5 44272054 IC50 = 5000 nM T65864 C0GEB5 44272057 IC50 = 163 nM T65864 C5AN1K 44272058 IC50 = 1400 nM T65864 CA7RU3 44272065 IC50 > 16700 nM T65864 COG91E 44272066 IC50 = 1000 nM T65864 C6G2YI 44272074 IC50 = 36 nM T65864 CL0CH1 44272075 IC50 > 16700 nM T65864 CHX4C2 44272087 IC50 = 123 nM T65864 C6J5NI 44272088 IC50 = 9800 nM T65864 C4O0CH 44272164 IC50 = 610 nM T65864 CX28HG 44272165 IC50 = 750 nM T65864 CJ2P4U 44272187 IC50 = 441 nM T65864 C8W1PC 44272190 IC50 = 5310 nM T65864 CLHI94 44272192 IC50 = 464 nM T65864 CNME25 44272315 IC50 = 663 nM T65864 CH9B3K 44272329 IC50 = 43 nM T65864 CPE46J 44272330 IC50 = 60 nM T65864 CVU8Y5 44272331 IC50 = 42 nM T65864 C9QU0A 44272339 IC50 = 660 nM T65864 CX1DC3 44272340 IC50 = 27 nM T65864 C25ZPQ 44286077 IC50 = 160 nM T65864 C2VT5D 44286078 IC50 = 110 nM T65864 C5TNF1 44286080 IC50 = 45 nM T65864 C6DQ8C 44286082 IC50 = 140 nM T65864 C56UNI 44286141 IC50 = 87 nM T65864 CP9Z6L 44286142 IC50 = 430 nM T65864 CG9MD1 44286153 IC50 = 57 nM T65864 C0Q4YT 44286175 IC50 = 37 nM T65864 C3X9OZ 44286176 IC50 = 69 nM T65864 CANQ14 44286178 IC50 = 35 nM T65864 CMYO82 44286192 IC50 = 420 nM T65864 C4O0NY 44286195 IC50 = 54 nM T65864 C2JUK5 44286295 IC50 = 38 nM T65864 CL42KC 44286313 IC50 = 70 nM T65864 C7TN9R 44286314 IC50 = 290 nM T65864 CD1W2V 44286325 IC50 = 69 nM T65864 CSN39H 44286341 IC50 = 33 nM T65864 C7U0FQ 44286342 IC50 = 310 nM T65864 CQM8T4 44286449 IC50 = 53 nM T65864 C3S7FL 44286458 IC50 = 235 nM T65864 CM1D0Y 44286459 IC50 = 183 nM T65864 CTE57J 44286514 IC50 = 200 nM T65864 CKHP61 44290243 IC50 = 310 nM T65864 CMH1I6 44304594 IC50 = 797 nM T65864 CQP25N 44304665 IC50 = 120 nM T65864 C3LI2Q 44304736 IC50 = 710 nM T65864 CEG4W3 44304738 IC50 = 2 nM T65864 CO97ZN 44304740 IC50 = 200 nM T65864 CM5LG0 44304767 IC50 = 220 nM T65864 CB2K6C 44304876 IC50 = 110 nM T65864 C9D3SY 44304908 IC50 > 500 nM T65864 CNS90X 44304987 IC50 = 260 nM T65864 CE93TR 44305012 IC50 = 325 nM T65864 C1K3XE 44305055 IC50 = 160 nM T65864 CD48GV 44323871 IC50 = 530 nM T65864 CTCE98 44324149 IC50 = 44 nM T65864 C6G2FS 44326041 IC50 = 25 nM T65864 C1J0EO 44327116 IC50 = 47 nM T65864 CMLC78 44327214 IC50 = 0.3 nM T65864 CBCA97 44327250 IC50 = 0.5998 nM T65864 C9MI7V 44327255 IC50 = 2.399 nM T65864 CCK31F 44327256 IC50 = 7 nM T65864 C1BN4R 44327272 IC50 = 0.4 nM T65864 CET82L 44327289 IC50 = 130 nM T65864 CW39RD 44327290 IC50 = 169.82 nM T65864 CI2Z9M 44327356 IC50 = 44 nM T65864 C8BV2G 44327372 IC50 = 320 nM T65864 CP0HW4 44327376 IC50 = 44 nM T65864 CO5J3A 44327391 IC50 = 11 nM T65864 CZJP98 44327394 IC50 = 22 nM T65864 C0SAO1 44327408 IC50 = 67 nM T65864 CC54QV 44327459 IC50 = 1.5 nM T65864 CM6DU7 44327473 IC50 = 0.13 nM T65864 C9Y3HI 44327474 IC50 = 0.1 nM T65864 CUX68M 44327477 IC50 = 0.1 nM T65864 CKAQ93 44327664 IC50 = 10.99 nM T65864 CT8IR5 44327665 IC50 = 79 nM T65864 C57RSX 44327685 IC50 = 7 nM T65864 CA7QD8 44327730 IC50 = 30 nM T65864 CZ3TW1 44328802 IC50 = 610 nM T65864 CFYC63 44328896 IC50 = 170 nM T65864 CS5M6I 44328970 IC50 = 42 nM T65864 CTU05A 44329036 IC50 = 53 nM T65864 CUSZ54 44329092 IC50 = 18 nM T65864 C3OL0J 44329237 IC50 = 390 nM T65864 C3CX4A 44335244 IC50 = 1540 nM T65864 CX28YN 44335417 IC50 = 1650 nM T65864 C8MP9H 44335468 IC50 = 1300 nM T65864 C3APV8 44339273 IC50 = 559 nM T65864 CWH5G9 44345925 IC50 = 11000 nM T65864 CQVW76 44346052 IC50 = 1800 nM T65864 C87MEG 44346063 IC50 > 20000 nM T65864 C2UAQ1 44351275 IC50 = 5400 nM T65864 CS8Y4I 44351755 IC50 = 80 nM T65864 CMXT47 44351792 IC50 = 1815 nM T65864 CDU6R5 44351815 IC50 = 100 nM T65864 CF1H6Y 44351831 IC50 = 80 nM T65864 CZF21R 44351880 IC50 = 38 nM T65864 CIEM10 44351882 IC50 = 36 nM T65864 CTB3W1 44351888 IC50 = 47 nM T65864 CMG81Z 44351899 IC50 = 54 nM T65864 C2NYO0 44351900 IC50 = 48 nM T65864 C4U0OX 44351906 IC50 = 600 nM T65864 CWV8P9 44351908 IC50 = 69 nM T65864 C8RQY2 44351909 IC50 = 66 nM T65864 CSG20K 44351945 IC50 = 96 nM T65864 CIK46B 44351950 IC50 = 110 nM T65864 C8U3MH 44351953 IC50 = 2190 nM T65864 C1VN5S 44351954 IC50 = 1850 nM T65864 CMJ9G4 44351956 IC50 = 1420 nM T65864 CUL6X2 44351971 IC50 = 32 nM T65864 CT4SH8 44351972 IC50 = 94 nM T65864 CLJ6P8 44351973 IC50 = 450 nM T65864 C7MHU6 44351974 IC50 = 260 nM T65864 CS61LI 44351984 IC50 = 350 nM T65864 CFL16M 44351990 IC50 = 200 nM T65864 C72EHI 44351994 IC50 = 49 nM T65864 C5G7JS 44351997 IC50 = 110 nM T65864 CQZ5B8 44352051 IC50 = 120 nM T65864 C5J0YM 44352052 IC50 = 270 nM T65864 C47DES 44352068 IC50 < 30 nM T65864 CY6ST1 44352069 IC50 = 16 nM T65864 CLG9R7 44352098 IC50 = 1990 nM T65864 C3PA0D 44352101 IC50 = 230 nM T65864 C6HN1F 44352102 IC50 = 180 nM T65864 C1BPA5 44352280 IC50 = 340 nM T65864 CQG9P3 44352281 IC50 = 113 nM T65864 C3I4MH 44368287 IC50 > 100000 nM T65864 CIMO40 44372376 IC50 = 90 nM T65864 CAD1P9 44372396 IC50 = 320 nM T65864 CZ6T1E 44372397 IC50 > 10000 nM T65864 CT8K9G 44372405 IC50 = 800 nM T65864 CRP9D1 44372406 IC50 = 180 nM T65864 CC6NH7 44372451 IC50 = 1000 nM T65864 CE5TI8 44372454 IC50 > 1000 nM T65864 C6VFJ4 44372477 IC50 > 10000 nM T65864 CE72TG 44372478 IC50 > 10000 nM T65864 C4QMX9 44372556 IC50 = 1230 nM T65864 CPZJ67 44372577 IC50 = 160 nM T65864 CXN20W 44372638 IC50 = 340 nM T65864 CW9A4U 44372650 IC50 = 2800 nM T65864 CU08DK 44372676 IC50 = 14200 nM T65864 CJ42WU 44372677 IC50 = 2650 nM T65864 CYNM09 44372688 IC50 = 2840 nM T65864 C0I9AX 44372700 IC50 = 1000 nM T65864 C36GFB 44372701 IC50 = 300 nM T65864 C0L8YS 44372720 IC50 = 1150 nM T65864 C3LP6U 44372846 IC50 = 1360 nM T65864 C7X0JK 44372847 IC50 = 1690 nM T65864 C14DKZ 44372856 IC50 > 10000 nM T65864 CFOC83 44372888 IC50 = 210 nM T65864 C6R7OP 44372904 IC50 = 5540 nM T65864 CU6O1J 44372923 IC50 = 2680 nM T65864 CPKI70 44372946 IC50 = 420 nM T65864 CER69Z 44373083 IC50 = 50 nM T65864 C0CBK8 44373103 IC50 = 260 nM T65864 CFEW63 44373192 IC50 = 3760 nM T65864 CQA71Y 44394686 IC50 = 320 nM T65864 C7A6ZC 44394687 IC50 = 460 nM T65864 C1DGX8 44394827 IC50 = 360 nM T65864 CZS4N7 44394840 IC50 = 11200 nM T65864 C2S4PW 44394843 IC50 = 280 nM T65864 C6OM1L 44394880 IC50 = 6600 nM T65864 C6BNY3 44394888 IC50 = 2200 nM T65864 C2EKR8 44395031 IC50 = 280 nM T65864 C8H9TQ 44395035 IC50 = 166 nM T65864 C8PG0K 44395041 IC50 = 90 nM T65864 CU9Z5Y 44395043 IC50 = 50 nM T65864 CF31XZ 44395044 IC50 = 10 nM T65864 CC9KY5 44395045 IC50 = 20 nM T65864 CZ7FY4 44395049 IC50 = 1220 nM T65864 CJ2XD8 44395051 IC50 = 40 nM T65864 C6MWZ0 44395075 IC50 = 450 nM T65864 C2F9YS 44395089 IC50 = 50 nM T65864 C0T2GL 44395101 IC50 = 50 nM T65864 CY9R4E 44395109 IC50 = 20 nM T65864 CLQ18K 44395115 IC50 = 50 nM T65864 CL27MX 44395117 IC50 > 20000 nM T65864 C1XWN9 44395122 IC50 = 90 nM T65864 CCLX29 44395123 IC50 = 690 nM T65864 C1INK2 44395139 IC50 = 100 nM T65864 C28BIC 44395140 IC50 = 60 nM T65864 CAQ2Z3 44395141 IC50 = 20 nM T65864 CCAI71 44395145 IC50 = 70 nM T65864 CXQJ50 44395146 IC50 = 90 nM T65864 CZ9WE4 44395151 IC50 = 230 nM T65864 CGNW80 44395161 IC50 = 20 nM T65864 CZ97PV 44395162 IC50 = 610 nM T65864 CNYD49 44395166 IC50 = 10 nM T65864 CZ6HP1 44395171 IC50 = 80 nM T65864 C2T6DH 44395178 IC50 = 40 nM T65864 CL8J9G 44395197 IC50 = 60 nM T65864 C2JV4I 44395203 IC50 = 20 nM T65864 C9KCD0 44395205 IC50 = 10 nM T65864 C28KMD 44395206 IC50 = 50 nM T65864 C0XQ2Z 44395209 IC50 = 210 nM T65864 CVY47N 44395233 IC50 = 50 nM T65864 CECF74 44395240 IC50 = 10 nM T65864 CTDI68 44395241 IC50 = 30 nM T65864 C0MT1L 44395257 IC50 = 10 nM T65864 C6EA4M 44396101 IC50 > 20000 nM T65864 CH56RI 44404432 IC50 = 116 nM T65864 CUW89Z 44404434 IC50 = 54 nM T65864 CW8F3T 44404438 IC50 = 217 nM T65864 C9AJ1Y 44404441 IC50 = 31 nM T65864 C2RXS6 44404444 IC50 = 46 nM T65864 C2MT9X 44404797 IC50 = 3.2 nM T65864 CAC7Q5 44404813 IC50 = 3.981 nM T65864 CJK6L9 44405349 IC50 > 20000 nM T65864 C7KGZ1 44405350 IC50 > 20000 nM T65864 CAEW63 44405351 IC50 > 20000 nM T65864 C5Z3KX 44405372 IC50 > 20000 nM T65864 CZ2DC4 44405388 IC50 = 16000 nM T65864 CCT95H 44405389 IC50 > 20000 nM T65864 C5R2SZ 44405413 IC50 = 400 nM T65864 C0DG2U 44405438 IC50 = 10000 nM T65864 CINB75 44405449 IC50 = 1200 nM T65864 C8HV2Y 44405934 IC50 = 2.2 nM T65864 C4F6US 44405954 IC50 = 3.2 nM T65864 C53BPJ 44406000 IC50 = 3.2 nM T65864 C0XZ8K 44406013 IC50 > 20000 nM T65864 CS3K1P 44406014 IC50 > 20000 nM T65864 CC93JP 44406018 IC50 > 20000 nM T65864 CCRZ12 44406074 IC50 > 20000 nM T65864 C8B7MF 44406105 IC50 = 0.26 nM T65864 CK0G6Y 44408608 IC50 = 51000 nM T65864 C7F6KQ 44408641 IC50 = 251 nM T65864 CFY5E9 44408670 IC50 = 199 nM T65864 CI76KB 44408825 IC50 = 37 nM T65864 CBC3X6 44408908 IC50 = 50 nM T65864 CY8LJ5 44408909 IC50 = 162 nM T65864 C3O7GC 44408936 IC50 = 171 nM T65864 CCW09A 44408944 IC50 = 421 nM T65864 CXIU70 44412815 IC50 = 1000 nM T65864 CX1BF9 44412816 IC50 > 5000 nM T65864 CJAG02 44412824 IC50 = 1420 nM T65864 CQ0A5Y 44412830 IC50 > 5000 nM T65864 CO9W0C 44412831 IC50 = 6160 nM T65864 C1S2CL 44412844 IC50 > 5000 nM T65864 CEYO05 44412845 IC50 > 5000 nM T65864 C1PJ2L 44412988 IC50 = 3100 nM T65864 C43VIW 44412989 IC50 = 3650 nM T65864 CSJ09N 44413000 IC50 = 2880 nM T65864 CI0C8G 44413001 IC50 > 5000 nM T65864 CE8C9M 44413012 IC50 = 843 nM T65864 C8G5YN 44415111 IC50 = 3200 nM T65864 CHJ7T1 44415158 IC50 = 200 nM T65864 C5TQ4F 44415291 IC50 = 3000 nM T65864 CXR91C 44419745 IC50 = 11 nM T65864 C4DM0E 44421260 IC50 = 73 nM T65864 CW95OG 44421262 IC50 = 28 nM T65864 C12DAL 44421263 IC50 = 250 nM T65864 CH58GC 44421265 IC50 = 264 nM T65864 C2JC0U 44421268 IC50 = 346 nM T65864 C13PXR 44421270 IC50 = 100 nM T65864 C8OJ3C 44421275 IC50 = 53 nM T65864 CAF94I 44421276 IC50 = 227 nM T65864 CP32ZD 44421391 IC50 > 1000 nM T65864 CPBK03 44426947 IC50 = 97 nM T65864 CDK97Q 44426948 IC50 = 68 nM T65864 C5WK0J 44426949 IC50 = 112 nM T65864 CMI8O6 44426950 IC50 = 154 nM T65864 C4BA1K 44426951 IC50 = 55 nM T65864 CQ34EI 44426952 IC50 = 40 nM T65864 CGU72L 44426953 IC50 = 37 nM T65864 C6R4BA 44426954 IC50 = 40 nM T65864 C4UJ8P 44426955 IC50 = 30 nM T65864 C09ZFD 44426958 IC50 = 26 nM T65864 CX5TJ4 44426959 IC50 = 39 nM T65864 CA65UR 44426961 IC50 = 137 nM T65864 C6SA0N 44426963 IC50 = 593 nM T65864 C5X7GE 44426965 IC50 = 167 nM T65864 C50GXW 44426967 IC50 = 38 nM T65864 CLS3R8 44426970 IC50 = 50 nM T65864 C5A0EI 44426971 IC50 = 164 nM T65864 C9KR5G 44426974 IC50 = 13 nM T65864 CU0L5B 44426977 IC50 = 14 nM T65864 CZEQ79 44426980 IC50 = 13 nM T65864 C5DB8P 44426982 IC50 = 16 nM T65864 CD7MB9 44426997 IC50 = 195 nM T65864 C5YUK6 44431823 IC50 > 15848.93 nM T65864 CO91FC 44431824 IC50 > 15848.93 nM T65864 CI95TS 44431825 IC50 > 15848.93 nM T65864 CJN16A 44431826 IC50 > 15848.93 nM T65864 CU75OI 44431827 IC50 > 15848.93 nM T65864 C2P8TK 44431828 IC50 > 15848.93 nM T65864 C2C4SX 44431829 IC50 > 15848.93 nM T65864 C9Y1ID 44431830 IC50 > 15848.93 nM T65864 CU20ER 44431831 IC50 > 15848.93 nM T65864 CL87AX 44431832 IC50 > 15848.93 nM T65864 CA61VJ 44431833 IC50 > 15848.93 nM T65864 C1KW0V 44431834 IC50 > 15848.93 nM T65864 CLV47X 44447379 IC50 = 5200 nM T65864 C0ZI2V 44447384 IC50 = 2200 nM T65864 CB5W6M 44447388 IC50 = 3100 nM T65864 C7YAB2 44447403 IC50 = 9700 nM T65864 C62MQL 44447909 IC50 = 140 nM T65864 COZ7P1 44447910 IC50 = 28 nM T65864 CKGC10 44447911 IC50 = 13 nM T65864 CI9W8E 44447914 IC50 = 36 nM T65864 C2WGB7 44447926 IC50 = 270 nM T65864 C80DRL 44447927 IC50 = 110 nM T65864 CWG8N1 44447934 IC50 = 110 nM T65864 CE0N7I 44447935 IC50 = 160 nM T65864 CA95RG 44447936 IC50 = 34 nM T65864 C60EOJ 44447938 IC50 = 53 nM T65864 CW43TR 44447940 IC50 = 330 nM T65864 C8BT7N 44447941 IC50 = 130 nM T65864 CQ51GD 44448073 IC50 = 21 nM T65864 C4G7IQ 44448074 IC50 = 21 nM T65864 COQ32D 44448075 IC50 = 7.1 nM T65864 C4VS3R 44448076 IC50 > 1000 nM T65864 CFW1K9 44448077 IC50 = 33 nM T65864 CI8T7E 44448078 IC50 = 146 nM T65864 CJDS83 44448079 IC50 > 1000 nM T65864 CM7GQ0 44448080 IC50 = 72 nM T65864 CBU30X 44448081 IC50 = 175 nM T65864 CO85QC 44448082 IC50 = 48 nM T65864 C1IQD9 44448083 IC50 = 33 nM T65864 CA6SD5 44448084 IC50 = 20 nM T65864 CF27CQ 44448085 IC50 = 3.3 nM T65864 CC9B8K 44448086 IC50 = 47 nM T65864 C4TA9Y 44448087 IC50 = 16 nM T65864 C0N3OK 44448088 IC50 = 12 nM T65864 CV0U4J 44448089 IC50 = 6.5 nM T65864 C3JYC2 44448090 IC50 = 10 nM T65864 C1YN7X 44448091 IC50 = 1.6 nM T65864 C03BHW 44448092 IC50 = 2.7 nM T65864 CZ2A6L 44448093 IC50 = 3.7 nM T65864 CB43PA 44448094 IC50 = 5.5 nM T65864 C08OFM 44448095 IC50 = 11 nM T65864 CMKE63 44449750 Ki = 0.54 nM T65864 CTX1H5 44449752 IC50 = 23 nM T65864 C7K1SF 44449773 IC50 = 2 nM T65864 C5L9BI 44449797 IC50 = 5 nM T65864 C1Z9YW 44449801 IC50 = 5 nM T65864 CVM5X4 44449803 Ki = 0.42 nM T65864 CQW4P5 44449831 IC50 = 4 nM T65864 C7M2QL 44449832 IC50 = 3 nM T65864 CG73IQ 44449833 IC50 = 1 nM T65864 C5F4PZ 44449859 IC50 = 2 nM T65864 CB6D3U 44449886 IC50 = 16 nM T65864 C0W2JY 44449890 IC50 = 27 nM T65864 CRAB85 44449915 IC50 = 12 nM T65864 C3W5NS 44449917 IC50 = 23 nM T65864 CZ98BV 44449947 IC50 = 2 nM T65864 CSVJ48 44449948 IC50 = 16 nM T65864 CPFA49 44449949 IC50 = 7 nM T65864 C0PFC2 44449980 IC50 = 123 nM T65864 CD4P5X 44449981 IC50 = 924 nM T65864 CTY17N 44449982 Ki = 0.98 nM T65864 C0KV8H 44450008 IC50 = 14 nM T65864 C7G3HZ 44450009 Ki = 0.44 nM T65864 CCD41K 44450034 Ki = 3.4 nM T65864 CI0H3X 44450036 IC50 > 1000 nM T65864 CYZM17 44450063 IC50 = 13 nM T65864 C5OR8I 44450064 IC50 = 32 nM T65864 C4VU9G 44450065 IC50 > 1000 nM T65864 CYC7Z8 44450096 IC50 = 94 nM T65864 CZRN42 44450097 IC50 = 19 nM T65864 CL1KT8 44450106 IC50 = 8 nM T65864 C35KIY 44450138 IC50 = 240 nM T65864 C3JQ4R 44450163 IC50 = 10 nM T65864 C5XT9C 44450193 IC50 = 63 nM T65864 CH0CT1 44451687 IC50 > 1100 nM T65864 C5MQX7 44451688 IC50 > 1100 nM T65864 C8K5LD 44451690 IC50 > 1100 nM T65864 C0HY3S 44451713 IC50 > 1100 nM T65864 CN6D7M 44453140 IC50 = 130 nM T65864 C5WXI2 44453142 IC50 = 0.2 nM T65864 CZT52V 44453181 IC50 = 0.16 nM T65864 CTU03I 44453182 IC50 = 0.12 nM T65864 CAD15M 44453212 IC50 = 0.5 nM T65864 CZ87FI 44453244 IC50 = 0.3 nM T65864 CEOP52 44453245 IC50 = 1.5 nM T65864 CG75JF 44453276 IC50 = 0.9 nM T65864 CV5BT1 44453306 IC50 = 0.75 nM T65864 CWP46T 44453340 IC50 = 460 nM T65864 C4Y8SB 44453342 IC50 = 13.4 nM T65864 CVZL51 44453343 IC50 = 350 nM T65864 CWI86M 44453344 IC50 = 5 nM T65864 C7YZ0B 44453380 IC50 = 28 nM T65864 CZRB17 44453417 IC50 = 4 nM T65864 CNK08A 44453419 IC50 = 9 nM T65864 CW0CX3 44453448 IC50 = 6 nM T65864 C7CD6R 44453484 IC50 = 27.5 nM T65864 C6C0HQ 44453701 IC50 = 150 nM T65864 CDV6X9 44454507 IC50 = 254 nM T65864 C6SMY7 44454538 IC50 = 2720 nM T65864 CZI92T 44454651 IC50 = 2.4 nM T65864 CZC95J 44454731 IC50 > 10000 nM T65864 C8LA2Y 44455915 IC50 = 3.9 nM T65864 CHE10T 44455949 IC50 = 5.1 nM T65864 CY81XN 44455989 IC50 = 3.7 nM T65864 CX6RH8 44456060 IC50 = 6.4 nM T65864 CTY20A 44456062 IC50 = 4.5 nM T65864 CMR98Z 44456093 IC50 = 2.5 nM T65864 CYBE29 44456097 IC50 = 3.5 nM T65864 CAQ96J 44456130 IC50 = 6 nM T65864 CI7V8S 44456134 IC50 = 11.2 nM T65864 CS71WV 44456177 IC50 = 16.2 nM T65864 C7DWO2 44456179 IC50 = 56.4 nM T65864 CJ80DS 44456213 IC50 = 88.4 nM T65864 C8GJ9Q 44456218 IC50 = 2489 nM T65864 CK06LJ 44456257 IC50 = 156 nM T65864 CN2Z5L 44456294 IC50 = 8.5 nM T65864 C0K2GQ 44456441 IC50 = 2.3 nM T65864 C5Z1TA 44456445 IC50 = 3.6 nM T65864 CDR4L1 44456448 IC50 = 7.2 nM T65864 C2JI7E 44456491 IC50 = 7 nM T65864 C0UV2I 44456495 IC50 = 3.2 nM T65864 CQJR79 44456499 IC50 = 3.9 nM T65864 C67VXQ 44457503 IC50 = 78 nM T65864 CV1G4E 44462686 IC50 = 470 nM T65864 C5LR0U 44462687 IC50 = 290 nM T65864 C5YC8L 44462688 IC50 = 95 nM T65864 CSI8G7 44463594 IC50 = 36 nM T65864 C2XVG6 44463863 IC50 = 400 nM T65864 CVHT52 44463864 IC50 = 19 nM T65864 CN1MD8 44463865 IC50 = 4 nM T65864 C7N2AQ 44473101 IC50 > 1600 nM T65864 C4MG3F 44473102 IC50 > 1600 nM T65864 CA85NJ 44473103 IC50 > 1600 nM T65864 CFK1A5 44473625 IC50 = 1200 nM T65864 CS26QA 44473783 IC50 = 2400 nM T65864 CL1CM8 44476045 IC50 = 0.16 nM T65864 C0O1QV 44476046 IC50 = 0.4 nM T65864 CBE5K9 44476050 IC50 = 5 nM T65864 CSP6V7 44476133 IC50 = 1.2 nM T65864 C7WTC4 44476134 IC50 = 38 nM T65864 C29OCA 44477382 IC50 = 0.9 nM T65864 C9L3HQ 44477383 IC50 = 38 nM T65864 CK3GZ6 44477384 IC50 = 4 nM T65864 C7TK5E 44479928 Ki = 3.981 nM T65864 CR60VL 44479929 Ki = 12.59 nM T65864 C50KGQ 44479930 Ki = 100 nM T65864 CN6B9S 44479931 Ki = 125.89 nM T65864 CB1I8L 44479933 Ki = 10 nM T65864 CEF20J 44479934 Ki = 12.59 nM T65864 C0RYL8 44480178 Ki = 10 nM T65864 CO0XS2 44480180 Ki = 794.33 nM T65864 C42CKX 44480181 Ki = 15.85 nM T65864 CQE20D 44480441 Ki = 7.943 nM T65864 C78ALJ 44480442 Ki = 7.943 nM T65864 C2XW9P 44480443 Ki = 12.59 nM T65864 CT38MK 44480444 Ki = 6.31 nM T65864 C8AW6R 44517629 IC50 = 50 nM T65864 CX87OQ 44517630 IC50 = 5 nM T65864 C8DEF1 44517631 IC50 = 4 nM T65864 C4MCY5 44517632 IC50 = 11 nM T65864 CN53CQ 44517633 IC50 = 2 nM T65864 C9Y7QJ 44517634 IC50 = 2340 nM T65864 C9A1XK 44517635 IC50 = 109 nM T65864 C8YHF3 44517636 IC50 = 218 nM T65864 CU80BP 44517743 IC50 = 1.5 nM T65864 C72LGV 44532791 Ki = 270 nM T65864 C4WRN5 44541014 IC50 = 50 nM T65864 C3VRO9 44557921 IC50 > 10000 nM T65864 CF16QB 44560451 IC50 = 1750 nM T65864 C0U8DH 44560546 IC50 = 455 nM T65864 CN3I8C 44560547 IC50 = 24 nM T65864 C0M1FW 44560587 IC50 = 1730 nM T65864 C18JQN 44560588 IC50 = 45 nM T65864 CS8GY1 44560640 IC50 = 181 nM T65864 C6VF0N 44560641 IC50 = 57.8 nM T65864 C1CO0M 44565383 IC50 = 130 nM T65864 C5NFS4 44565384 IC50 = 95 nM T65864 CZW89U 44565411 IC50 = 2530 nM T65864 CIJ2Z4 44568178 IC50 > 1000 nM T65864 C29IYW 44568179 IC50 > 1000 nM T65864 CX45TP 44568180 IC50 > 1000 nM T65864 CPX96E 44568181 IC50 > 1000 nM T65864 C91EKS 44568215 IC50 > 1000 nM T65864 CKO23U 44568218 IC50 = 960 nM T65864 CU52QC 44568219 IC50 = 70 nM T65864 C0MIN7 44568220 IC50 = 42 nM T65864 CLJ0T1 44568221 IC50 = 235 nM T65864 CW8T5V 44568222 IC50 = 38 nM T65864 C9MZT3 44568225 IC50 = 146 nM T65864 CF3UX6 44568254 IC50 = 424 nM T65864 CP5JA6 44568257 IC50 = 610 nM T65864 CY4LT0 44568258 IC50 = 40 nM T65864 CAE1R3 44568259 IC50 = 51 nM T65864 COX1A9 44568260 IC50 = 359 nM T65864 COC0F8 44568261 IC50 = 3 nM T65864 C8BT2D 44568262 IC50 = 211 nM T65864 C6J3BE 44568263 IC50 = 485 nM T65864 CTM0K2 44568298 IC50 = 191 nM T65864 CGEA32 44568299 IC50 = 140 nM T65864 CF16ZR 44568300 IC50 = 62.6 nM T65864 C0OD3P 44568332 IC50 = 260 nM T65864 CZT3F9 44568333 IC50 = 87.1 nM T65864 CIWL70 44568334 IC50 = 859 nM T65864 CR53DN 44568335 IC50 = 344 nM T65864 CN43BI 44568359 IC50 = 55.1 nM T65864 C4M1SH 44568360 IC50 = 225 nM T65864 CES3O1 44568361 IC50 = 55.6 nM T65864 CW52NV 44568386 IC50 = 916 nM T65864 CSCY70 44568387 IC50 = 148 nM T65864 CC7MB2 44568388 IC50 = 28 nM T65864 CL95CO 44568389 IC50 = 95.4 nM T65864 CZMX10 44568412 IC50 = 54.4 nM T65864 CIXK10 44568413 IC50 = 62.8 nM T65864 C5HRV7 44568414 IC50 = 78 nM T65864 CCH60W 44568463 IC50 = 48.5 nM T65864 CB2Q6R 44568681 IC50 = 411 nM T65864 C3SQE6 44568682 IC50 = 213 nM T65864 C8IOV0 44568683 IC50 = 372 nM T65864 C16NYL 44568698 IC50 > 1000 nM T65864 C2EXW6 44568699 IC50 > 1000 nM T65864 C56GCD 44568700 IC50 > 1000 nM T65864 C9N3UM 44568701 IC50 > 1000 nM T65864 C3OP7X 44568735 IC50 = 657 nM T65864 CP59GK 44568736 IC50 = 1950 nM T65864 CZMG67 44568751 IC50 > 1000 nM T65864 C0EI3M 44568752 IC50 > 1000 nM T65864 C7CH4M 44568753 IC50 > 1000 nM T65864 C03JAH 44568754 IC50 > 1000 nM T65864 CJB91U 44568803 Ki = 0.4 nM T65864 CR7C6A 44568804 Ki = 0.7 nM T65864 C97CEZ 44568805 Ki = 2 nM T65864 CQ7SL3 44568819 Ki = 0.8 nM T65864 C1OVN0 44568820 Ki = 0.5 nM T65864 C4MNS3 44568821 Ki = 0.3 nM T65864 COPU28 44568925 Ki = 1.1 nM T65864 CSQ1F7 44568926 Ki = 0.3 nM T65864 C6QG1U 44568927 Ki = 0.4 nM T65864 CT2CX7 44568928 Ki = 0.6 nM T65864 CCV6K0 44568929 Ki = 0.2 nM T65864 C25LHW 44568941 Ki = 0.5 nM T65864 CK67DM 44568942 Ki = 0.2 nM T65864 C3PTD5 44568943 Ki = 0.4 nM T65864 C4CX6W 44568944 Ki = 0.3 nM T65864 C1LGP4 44568945 Ki = 16 nM T65864 CX4HV8 44570785 EC50 = 28100 nM T65864 CJ63ZW 44570787 EC50 = 13530 nM T65864 C9NHM1 44570788 EC50 = 15000 nM T65864 CB19GI 44571327 EC50 = 14830 nM T65864 CL5ZS4 44571329 EC50 = 10900 nM T65864 CP38YF 44571362 EC50 = 14200 nM T65864 C9TA0K 44571363 EC50 = 41200 nM T65864 CWF4P5 44571364 IC50 = 12500 nM T65864 CHK7O0 44571365 EC50 = 22000 nM T65864 CKE8N1 44571813 IC50 = 9 nM T65864 CWFB42 44571820 IC50 = 1800 nM T65864 CEFU41 44572271 IC50 = 740 nM T65864 CCL85F 44575073 IC50 = 21660 nM T65864 CJX06P 44575126 IC50 > 50000 nM T65864 CE8FC7 44575127 IC50 > 50000 nM T65864 CR2VB0 44577779 IC50 = 0.7 nM T65864 CJ6P3H 44578238 Ki = 730 nM T65864 C62SFQ 44578252 Ki = 430 nM T65864 CSO67T 44578253 Ki = 1400 nM T65864 CF7H1U 44578254 Ki = 400 nM T65864 C9QI5O 44578255 Ki = 130 nM T65864 COL38H 44578306 Ki = 14 nM T65864 CC0F3Z 44578400 Ki = 630 nM T65864 CS27YJ 44578401 Ki = 170 nM T65864 C7I5HD 44578402 Ki = 350 nM T65864 C0IKS3 44578403 Ki = 40 nM T65864 C0BD8N 44578425 Ki = 70 nM T65864 CE1TR6 44578426 Ki = 330 nM T65864 CHG84Y 44578427 Ki = 1100 nM T65864 CVQK15 44578428 Ki = 1900 nM T65864 C08ECI 44578458 Ki = 25 nM T65864 C0ZHM6 44578459 Ki = 32 nM T65864 C4W0GN 44578460 Ki = 5 nM T65864 CJG7R1 44578461 Ki = 6 nM T65864 CWT38I 44578498 Ki = 5 nM T65864 C46QIA 44578499 Ki = 7 nM T65864 CY3KQ2 44578500 Ki = 4 nM T65864 CI1P7C 44578532 Ki = 3 nM T65864 C3QV8A 44578533 Ki = 43 nM T65864 CNF61D 44578534 Ki = 100 nM T65864 CLV20U 44578535 IC50 = 230 nM T65864 CEV86L 44578563 Ki > 2500 nM T65864 CP9T8W 44578564 Ki = 25 nM T65864 C0UO4C 44578565 Ki = 520 nM T65864 C8ESF0 44578566 Ki = 460 nM T65864 CN79GK 44578567 Ki = 940 nM T65864 CK52AC 44578612 Ki = 10 nM T65864 C79BYL 44578613 Ki > 2500 nM T65864 C4XGH5 44578614 Ki > 2500 nM T65864 CP8MD1 44578630 Ki = 300 nM T65864 C98WQP 44578670 Ki = 150 nM T65864 C71FZL 44578671 Ki = 14 nM T65864 CP6TG4 44578672 Ki = 1.9 nM T65864 C9VXN3 44578709 IC50 = 2 nM T65864 C4UY2L 44578710 Ki = 15 nM T65864 C2NXM3 44578711 Ki = 5.2 nM T65864 CKA4H9 44578746 Ki = 6.3 nM T65864 CD6M3G 44578747 Ki = 4.6 nM T65864 C65ZGB 44578748 Ki = 0.6 nM T65864 CZI74F 44578749 Ki = 3 nM T65864 C6LI5H 44578804 Ki = 100 nM T65864 CCR8P6 44578805 Ki = 2.1 nM T65864 C0IMF8 44578806 Ki = 1.6 nM T65864 CFT4G8 44578818 Ki = 20 nM T65864 CL1O8N 44578832 Ki = 11 nM T65864 C9DY0U 44578833 Ki = 79 nM T65864 CHT53L 44578843 Ki = 100 nM T65864 C3SR0I 44578844 Ki = 150 nM T65864 C3XQE9 44578845 Ki = 1600 nM T65864 C7Q1VU 44580077 Ki = 0.8 nM T65864 CY28MQ 44580283 Ki > 2000 nM T65864 CL90SE 44580358 Ki > 850 nM T65864 CF8RE4 44580359 Ki = 98 nM T65864 CI1M5E 44580360 Ki = 1.1 nM T65864 CNX70E 44580419 Ki > 850 nM T65864 CK1VE7 44580420 Ki = 2.8 nM T65864 CH2R7X 44580449 Ki = 1400 nM T65864 CY4U7D 44580489 Ki = 18 nM T65864 CN5LR7 44580490 Ki = 19 nM T65864 CZ4BC3 44580491 Ki = 11 nM T65864 CQC10N 44580531 Ki = 2000 nM T65864 C1VH0C 44580532 Ki = 6 nM T65864 CMI9D1 44580533 Ki = 6.7 nM T65864 C13AQY 44580534 Ki = 290 nM T65864 C7SQ6R 44580580 Ki = 49 nM T65864 C9IN8L 44580581 Ki > 2500 nM T65864 C6MYD1 44580582 Ki = 420 nM T65864 CY7B3E 44580583 Ki = 18 nM T65864 CRP13I 44580647 Ki = 2.4 nM T65864 C2CV6H 44580648 Ki > 2500 nM T65864 CXC52J 44580649 Ki = 11 nM T65864 CU7W9J 44580650 Ki = 4.5 nM T65864 CE32BQ 44580689 Ki = 830 nM T65864 C8D5IM 44580690 Ki = 490 nM T65864 CY80EG 44580691 Ki > 2500 nM T65864 C27ALZ 44580692 Ki = 1100 nM T65864 CMSR35 44580729 Ki = 380 nM T65864 CCU9A5 44580730 Ki = 160 nM T65864 CJR50B 44580731 Ki = 110 nM T65864 C93YSO 44580776 Ki = 19 nM T65864 CA31VJ 44580777 Ki = 12 nM T65864 C8Z5AX 44580778 Ki > 850 nM T65864 C9DO6G 44588777 IC50 = 14 nM T65864 CB4H1L 44588778 IC50 = 22 nM T65864 C7ZRO9 44588779 IC50 = 20 nM T65864 CC2S8A 44589676 IC50 = 150 nM T65864 C5Z3LI 44591740 IC50 = 15000 nM T65864 COY57J 44592504 IC50 = 25000 nM T65864 CY1A7W 44593407 IC50 = 219 nM T65864 C0QR1V 44593521 IC50 = 5 nM T65864 CO56GY 44593637 Ki = 70 nM T65864 CR76UZ 44593639 Ki = 12 nM T65864 CDC2V8 44593640 Ki = 6 nM T65864 CQ14ML 44593646 Ki = 1.9 nM T65864 CV8F0R 44593854 IC50 > 10000 nM T65864 C01TKN 44597013 IC50 = 30 nM T65864 C2RY3H 44597108 IC50 = 60 nM T65864 CMST74 44597109 IC50 = 450 nM T65864 CFD21J 44597110 IC50 = 6 nM T65864 CS7M8K 44597113 IC50 = 1560 nM T65864 CZ49BI 44597224 IC50 = 890 nM T65864 C6ET3K 44597225 IC50 = 2520 nM T65864 C7D8ZN 44597226 IC50 = 19 nM T65864 C4HN5F 44597227 IC50 = 41 nM T65864 C28QLM 44605035 IC50 = 28900 nM T65864 C75XHS 44605037 IC50 > 50000 nM T65864 CH3SF9 44631836 Ki = 1 nM T65864 CNX84R 44817010 IC50 = 11000 nM T65864 C61HBG 45102725 IC50 = 200 nM T65864 CVED60 45254198 IC50 = 1 nM T65864 C53MQJ 45254575 IC50 = 31 nM T65864 CS9Y8K 45254577 IC50 = 6 nM T65864 CNJY05 45256216 IC50 = 8 nM T65864 C7YCA2 45257074 IC50 = 2 nM T65864 C19HUI 45257075 IC50 = 2 nM T65864 C8QZ0C 45267493 IC50 > 1000 nM T65864 C2W8KF 45267518 IC50 = 6.1 nM T65864 CTEG46 45268375 IC50 = 1.2 nM T65864 CY12WO 45268376 IC50 = 4 nM T65864 C6B7WN 45268386 IC50 = 13 nM T65864 CVX26E 45268398 IC50 = 1.4 nM T65864 CA23MC 45269229 IC50 = 8.5 nM T65864 CUXD21 45269245 IC50 = 1.1 nM T65864 CC96LP 45269578 IC50 > 10000 nM T65864 C19ANK 45270078 IC50 > 1000 nM T65864 C2SP4L 45270079 IC50 = 3.7 nM T65864 CLP20Q 45270908 IC50 > 1000 nM T65864 C0KJP8 45270909 IC50 = 2.6 nM T65864 CFT8P5 45271243 IC50 > 10000 nM T65864 C2BXF5 45271244 IC50 > 10000 nM T65864 CMT5Z2 45271247 IC50 > 10000 nM T65864 C1B0GM 45271770 IC50 = 1.1 nM T65864 C4JY6P 45272621 IC50 = 444 nM T65864 CM3S9C 45272627 IC50 = 1.1 nM T65864 C93DPH 45272642 IC50 = 7.8 nM T65864 CIY0D1 45272652 IC50 = 1.9 nM T65864 CTE15D 45272980 IC50 > 10000 nM T65864 CKT3S0 45273524 IC50 > 1000 nM T65864 CR4Y3E 45273538 IC50 = 269 nM T65864 CH2Q1I 45273565 IC50 = 3.3 nM T65864 CNRP95 45273566 IC50 = 1.9 nM T65864 CH31SM 45279906 IC50 = 20 nM T65864 C8MA3S 45279907 IC50 = 560 nM T65864 CE3X9A 45279908 IC50 = 140 nM T65864 C6IZ8R 45279909 IC50 = 60 nM T65864 CJY2F9 45279910 IC50 = 26700 nM T65864 COL2S0 45279912 IC50 = 8 nM T65864 CW4I0P 45279963 IC50 = 5 nM T65864 CFKE36 45279964 IC50 = 170 nM T65864 CJE1L5 45279965 IC50 = 20 nM T65864 CRX49V 45280411 IC50 = 40 nM T65864 C7KT8F 45280412 IC50 = 44 nM T65864 CYL0M9 45280413 IC50 = 40 nM T65864 CET20H 45280465 IC50 = 400 nM T65864 C3SYV8 45280466 IC50 = 70 nM T65864 C5E4VD 45280467 IC50 = 380 nM T65864 CMSY69 45280468 IC50 = 40 nM T65864 CGU65H 45280469 IC50 = 900 nM T65864 C2J3FM 45280530 IC50 = 10 nM T65864 CIK85S 45280531 IC50 = 10 nM T65864 C95KEU 45280584 IC50 = 20 nM T65864 CSZQ07 45280585 IC50 = 10400 nM T65864 CYK80Q 45280586 IC50 = 80 nM T65864 CXIB19 45280587 IC50 = 6000 nM T65864 C2K1BZ 45280638 IC50 = 20 nM T65864 CHRE26 45280639 IC50 = 20 nM T65864 CS2ZK0 45280640 IC50 = 80 nM T65864 CWS3L6 45280641 IC50 = 80 nM T65864 C4KU7J 45280642 IC50 = 440 nM T65864 CNV3L9 45280643 IC50 = 100000 nM T65864 CDJ7X4 45280692 IC50 = 158000 nM T65864 C6ENK8 45280693 IC50 = 40 nM T65864 C96GKZ 45280695 IC50 = 30 nM T65864 C2ZHY1 45280748 IC50 = 60 nM T65864 CZ8V9E 45280749 IC50 = 560 nM T65864 CC95PQ 45375865 IC50 > 50000 nM T65864 CEOQ27 45375866 IC50 > 50000 nM T65864 C6E2SC 45482700 IC50 > 10000 nM T65864 CZXH74 45482750 IC50 > 10000 nM T65864 C7BUV6 45486286 IC50 = 230 nM T65864 C6CP1M 45486287 IC50 = 140 nM T65864 C6OQS0 45486309 IC50 = 1100 nM T65864 CQK6E0 45487937 IC50 = 370 nM T65864 CA06GW 45487959 IC50 = 299 nM T65864 CUMF37 45487992 IC50 = 110 nM T65864 CFE79C 45487997 IC50 = 15 nM T65864 C46MWH 45488127 IC50 = 81 nM T65864 C97CXH 45488129 IC50 = 1380 nM T65864 C7R4NV 45488132 IC50 = 790 nM T65864 CK5AF2 45488133 IC50 = 1590 nM T65864 CP85DN 45488135 IC50 = 576 nM T65864 CD7M4K 45488136 IC50 = 9460 nM T65864 C9NBZ5 45488137 IC50 = 595 nM T65864 CRNQ39 45488140 IC50 = 259 nM T65864 CJDC01 45488141 IC50 = 608 nM T65864 CEF71R 45488144 IC50 = 114 nM T65864 C3P8YT 45488146 IC50 = 3150 nM T65864 CW9UX0 45488147 IC50 = 642 nM T65864 C6M3FY 45488148 IC50 = 211 nM T65864 CWU69I 45488149 IC50 = 238 nM T65864 CYEJ96 45488153 IC50 = 720 nM T65864 CBJ71F 45488154 IC50 = 3190 nM T65864 CLZ42E 45488157 IC50 = 1530 nM T65864 CGP15V 45488158 IC50 = 412 nM T65864 C1A5TZ 45488159 IC50 = 38 nM T65864 C7MB9G 45488160 IC50 = 333 nM T65864 C92NYI 45488168 IC50 = 3700 nM T65864 CWP89M 45488170 IC50 = 4790 nM T65864 CU9Y5O 45488173 IC50 = 6140 nM T65864 C3NCK5 45488177 IC50 = 431 nM T65864 CCD7O2 45892797 IC50 = 1230 nM T65864 C6FKV7 45910662 IC50 = 28330 nM T65864 C96BNW 46179972 IC50 > 50000 nM T65864 C38SHC 46182955 IC50 = 2.7 nM T65864 C9MR8B 46182956 IC50 = 2.7 nM T65864 C6WGB8 46182957 IC50 = 1.4 nM T65864 CD2LM3 46182958 IC50 = 2.6 nM T65864 C2QC0S 46184146 IC50 = 14.5 nM T65864 C9CJP7 46184147 IC50 = 2.7 nM T65864 CGS78K 46185428 IC50 = 0.9 nM T65864 CCL1U2 46185430 IC50 = 78 nM T65864 C34GUE 46185678 IC50 = 8.4 nM T65864 CGV57S 46185682 IC50 = 2.2 nM T65864 CXQI68 46197138 Ki = 458 nM T65864 CPGO35 46197139 Ki = 2 nM T65864 CY08KN 46197238 Ki = 2.3 nM T65864 CSN13Q 46197239 Ki = 8 nM T65864 C39BNV 46200949 IC50 = 100.2 nM T65864 CQJ7Z5 46200950 IC50 = 11 nM T65864 C89IVD 46201081 IC50 = 16 nM T65864 CUA97D 46209401 IC50 = 600 nM T65864 C03RVJ 46216734 IC50 = 9 nM T65864 CO5GE6 46225362 IC50 > 10000 nM T65864 CZT7C0 46225363 IC50 = 7370 nM T65864 CBM6P3 46226940 IC50 = 28.3 nM T65864 C6G8EB 46226943 IC50 = 7.2 nM T65864 CF9J6K 46226944 IC50 = 889 nM T65864 CDH2A5 46226945 IC50 = 3380 nM T65864 CZUO02 46226949 IC50 = 106 nM T65864 C6UYI8 46226951 IC50 = 1050 nM T65864 CLST29 46226954 IC50 = 322 nM T65864 C1VG8W 46226957 IC50 = 3770 nM T65864 CS4G8X 46226960 IC50 = 1170 nM T65864 CJ4LB9 46226962 IC50 = 141 nM T65864 CPYV78 46226969 IC50 = 33.3 nM T65864 CGR7M6 46226971 IC50 = 2920 nM T65864 CR09UC 46226973 IC50 = 8240 nM T65864 CAI7L4 46227810 IC50 = 16.3 nM T65864 CC67VM 46227813 IC50 = 79.3 nM T65864 C5Q6GU 46227816 IC50 = 24.9 nM T65864 C2P9QO 46228508 IC50 = 152 nM T65864 C6E5PY 46228822 IC50 = 1500 nM T65864 C3T8AM 46228951 IC50 = 608 nM T65864 C6Q4RS 46229583 IC50 = 405.2 nM T65864 CI4CT5 46229584 IC50 = 1648 nM T65864 CA0DS9 46229609 IC50 = 48.8 nM T65864 C0Y7GI 46229610 IC50 = 60.1 nM T65864 C4D7XZ 46229611 IC50 = 94.4 nM T65864 C4WT6O 46229612 IC50 = 105.2 nM T65864 CO1UY9 46229613 IC50 = 468.4 nM T65864 CS1IQ8 46229637 IC50 = 96.3 nM T65864 C5MP7O 46230872 IC50 > 10000 nM T65864 CFE9H3 46230873 IC50 = 100 nM T65864 C3M6RD 46230925 IC50 = 600 nM T65864 CJZA45 46232267 IC50 > 100000 nM T65864 C3PLE6 46232269 IC50 > 100000 nM T65864 C3U8HV 46232270 IC50 > 100000 nM T65864 CYA73D 46232312 IC50 > 100000 nM T65864 C54EKP 46232500 IC50 = 6 nM T65864 CRJV69 46232501 IC50 = 24 nM T65864 CB9QA4 46232502 IC50 = 29 nM T65864 C64LMQ 46232540 IC50 = 183 nM T65864 C3X9LS 46232541 IC50 = 47 nM T65864 C7EGB9 46232542 IC50 = 48 nM T65864 C9JE6X 46830346 IC50 = 100 nM T65864 CX8MJ9 46836027 IC50 = 3 nM T65864 CS8NX0 46836043 IC50 = 52 nM T65864 C0G1BS 46837667 IC50 = 23 nM T65864 CQ1R8K 46838229 IC50 = 49 nM T65864 C6KEH2 46838230 IC50 = 324 nM T65864 C9Y1ZW 46838231 IC50 = 468 nM T65864 CAK8W5 46864262 IC50 = 7 nM T65864 CQ78XK 46865783 IC50 = 3.3 nM T65864 CJ1V6W 46865784 IC50 = 1.7 nM T65864 C09BOA 46865979 IC50 = 19 nM T65864 CWY15J 46866401 IC50 = 54 nM T65864 CO1IG5 46866402 IC50 = 4 nM T65864 CO3P0J 46866604 IC50 < 50000 nM T65864 CW2G7D 46868853 IC50 > 50000 nM T65864 CR57OZ 46868855 IC50 > 5000 nM T65864 CI8YE5 46868856 IC50 > 50000 nM T65864 C94EPL 46868925 IC50 > 50000 nM T65864 C0GU4D 46868930 IC50 > 50000 nM T65864 CEK2I5 46869149 IC50 > 50000 nM T65864 C1VZM6 46869673 IC50 > 50000 nM T65864 CYI69K 46869674 IC50 > 50000 nM T65864 CSL2N6 46869740 IC50 > 50000 nM T65864 C6V9CD 46869741 IC50 > 50000 nM T65864 CZCQ05 46869742 IC50 > 50000 nM T65864 C09GAW 46869745 IC50 > 50000 nM T65864 CVBG98 46869815 IC50 > 5000 nM T65864 CU2D5N 46869816 IC50 > 50000 nM T65864 C8WH7Q 46869817 IC50 > 50000 nM T65864 CFOX43 46869876 IC50 > 5000 nM T65864 C2DW6T 46869878 IC50 > 50000 nM T65864 C19DQG 46869879 IC50 > 50000 nM T65864 CR1OH0 46869880 IC50 > 50000 nM T65864 CD1YH9 46869882 IC50 > 20000 nM T65864 C9KS6Q 46870032 IC50 = 27 nM T65864 C4MKC5 46870033 IC50 = 11 nM T65864 C5WC9K 46871765 IC50 = 540 nM T65864 CJOM49 46880136 IC50 = 69 nM T65864 C0X9HL 46880267 IC50 = 2.1 nM T65864 C4ZT9L 46880268 IC50 = 1.7 nM T65864 CCVM23 46880269 IC50 = 3 nM T65864 CS4JI7 46880311 IC50 = 4.1 nM T65864 CRI2V4 46880312 IC50 = 2.3 nM T65864 C34OCA 46880313 IC50 = 7.7 nM T65864 C2O3ZN 46880314 IC50 = 2.7 nM T65864 CRO4Z2 46880343 IC50 = 10 nM T65864 CE09XH 46880344 IC50 = 1.6 nM T65864 C9X8WS 46880345 IC50 = 6.3 nM T65864 C35PWX 46880869 IC50 = 1.6 nM T65864 C4ESF2 46880870 IC50 = 4.6 nM T65864 C01SRU 46880916 IC50 = 5 nM T65864 CNS7K6 46880917 IC50 = 8.5 nM T65864 CD5LH6 46880918 IC50 = 12 nM T65864 CLF48K 46880919 IC50 = 3 nM T65864 C5TAI0 46880957 IC50 = 43 nM T65864 C31BQI 46880958 IC50 = 10 nM T65864 CTS5Z1 46880959 IC50 = 36 nM T65864 C6WD4Q 46881329 IC50 > 15848.93 nM T65864 C6GQH3 46881341 IC50 > 15848.93 nM T65864 CEK6A9 46881342 IC50 > 15848.93 nM T65864 C84TWY 46881343 IC50 > 15848.93 nM T65864 C1DFI0 46881344 IC50 > 15848.93 nM T65864 CW32UX 46881345 IC50 > 15848.93 nM T65864 C8CE7P 46881351 IC50 > 15848.93 nM T65864 C7AE4V 46881352 IC50 > 15848.93 nM T65864 CP7UE5 46881353 IC50 > 15848.93 nM T65864 C32XZI 46881354 IC50 > 15848.93 nM T65864 CSQ8O9 46881355 IC50 > 15848.93 nM T65864 CO0SC4 46881358 IC50 > 15848.93 nM T65864 C4DXW0 46881359 IC50 = 12589.25 nM T65864 CK67BQ 46881360 IC50 > 15848.93 nM T65864 CV4O5T 46881361 IC50 > 15848.93 nM T65864 CHU3Z8 46882355 IC50 = 200 nM T65864 CZ47SV 46882356 IC50 = 25 nM T65864 CSH38Q 46882357 IC50 = 1000 nM T65864 C6Z0YR 46882358 IC50 = 380 nM T65864 C5NG6O 46882404 IC50 = 390 nM T65864 CSX7Y1 46882405 IC50 = 150 nM T65864 CRQ5E3 46882406 IC50 = 210 nM T65864 C1C0YG 46882407 IC50 = 450 nM T65864 C2KMV1 46882408 IC50 = 450 nM T65864 CZ15LR 46882469 IC50 = 180 nM T65864 CRD8S3 46884198 IC50 = 54 nM T65864 CYQ25D 46884595 IC50 = 99.6 nM T65864 CXC97Z 46884596 IC50 = 67.3 nM T65864 CS3UI6 46884597 IC50 = 41 nM T65864 CY3T2E 46884634 IC50 = 106 nM T65864 CQH28F 46884635 IC50 = 14 nM T65864 CQ7E0D 46884636 IC50 = 126 nM T65864 CIT8B5 46884665 IC50 = 111 nM T65864 CT6Y1E 46884695 IC50 = 184 nM T65864 C1EY3N 46884696 IC50 = 31 nM T65864 CNH51B 46884697 IC50 = 205 nM T65864 CC6BE5 46884730 IC50 = 47 nM T65864 CET05C 46884779 IC50 = 88 nM T65864 C84NWT 46886049 IC50 = 1110 nM T65864 C81VXS 46886050 IC50 = 65 nM T65864 CB41AU 46886051 IC50 = 104 nM T65864 CF0TX6 46886052 IC50 = 64 nM T65864 CW7NO2 46886053 IC50 = 39 nM T65864 COZF65 46886054 IC50 = 26 nM T65864 C7RL4A 46886114 IC50 = 462 nM T65864 C24PEO 46886115 IC50 = 165 nM T65864 CB2S4M 46886116 IC50 = 345 nM T65864 C5R7AJ 46886117 IC50 = 158 nM T65864 CT3Q6W 46886132 IC50 > 10000 nM T65864 COA0G1 46886133 IC50 > 10000 nM T65864 C9BH2Q 46886134 IC50 = 711 nM T65864 CT1HS5 46886166 IC50 = 673 nM T65864 CJ8S1K 46886167 IC50 > 10000 nM T65864 CIL51G 46886168 IC50 = 96 nM T65864 CYXW48 46886190 IC50 = 72 nM T65864 CFQ8U3 46886191 IC50 = 24 nM T65864 COP67X 46886192 IC50 = 360 nM T65864 CT4J3C 46886193 IC50 = 400 nM T65864 CHZ87M 46886218 IC50 = 316 nM T65864 C1E2WO 46886219 IC50 = 3040 nM T65864 CP8V4W 46886220 IC50 = 600 nM T65864 CK7D6Y 46886246 IC50 = 17 nM T65864 CSD79I 46886247 IC50 = 11 nM T65864 CT43QU 46886248 IC50 = 25 nM T65864 CZ90FU 46886249 IC50 = 310 nM T65864 C4MH2G 46886449 IC50 = 64 nM T65864 CVC86S 46886450 IC50 = 17 nM T65864 C8HOD9 46886476 IC50 = 7800 nM T65864 CYG1P8 46886477 IC50 = 164 nM T65864 CP1WS4 46886478 IC50 = 71 nM T65864 CFC3J0 46886479 IC50 = 90 nM T65864 C42GOJ 46886480 IC50 = 45 nM T65864 C0QX6T 46886481 IC50 = 180 nM T65864 C8MN3J 46886500 IC50 = 589 nM T65864 C7F1JP 46886501 IC50 = 408 nM T65864 C4FTH7 46886502 IC50 = 188 nM T65864 CW03LG 46886503 IC50 = 154 nM T65864 C7BT8N 46886504 IC50 = 179 nM T65864 C74PKJ 46886505 IC50 = 193 nM T65864 C38XWB 46886506 IC50 = 267 nM T65864 CX1P7Q 46886530 IC50 = 7540 nM T65864 C5Q3JK 46886531 IC50 = 81 nM T65864 C4T3VQ 46886532 IC50 = 313 nM T65864 C0TBQ2 46886533 IC50 = 13 nM T65864 CMN15K 46886534 IC50 = 91 nM T65864 C87FNK 46886535 IC50 = 81 nM T65864 C0E6XI 46887066 IC50 > 100000 nM T65864 CNQM15 46887067 IC50 = 24400 nM T65864 C7VGU9 46887068 IC50 = 2700 nM T65864 C0JQ8T 46887097 IC50 = 1390 nM T65864 C5LAW7 46887098 IC50 = 5720 nM T65864 CM6CO3 46887099 IC50 = 3140 nM T65864 CT78EQ 46887100 IC50 = 3810 nM T65864 C38LYC 46887134 IC50 = 12300 nM T65864 C6JEI1 46887135 IC50 = 540 nM T65864 C6L1VH 46887136 IC50 = 470 nM T65864 C2WM7V 46887184 IC50 = 1010 nM T65864 C1VZ0G 46887185 IC50 = 590 nM T65864 C3O8AM 46887186 IC50 = 15 nM T65864 CZ7M4V 46919120 IC50 = 18.4 nM T65864 C5WBZ7 46919121 IC50 = 1 nM T65864 CNL40R 46919122 IC50 = 189.3 nM T65864 CN8T1A 46919703 IC50 = 21 nM T65864 C60GAV 46929544 IC50 = 8000 nM T65864 C2QZ1I 46930629 IC50 = 328 nM T65864 C9VFU0 46930630 IC50 = 111 nM T65864 CB51LJ 46930631 IC50 = 299 nM T65864 CX0G7W 46930632 IC50 = 55.8 nM T65864 CMF1N8 46930633 IC50 = 6.1 nM T65864 CQB3E1 46930634 IC50 > 1000 nM T65864 CQY80A 46930726 IC50 = 3.1 nM T65864 CQR9K1 46933384 IC50 > 100000 nM T65864 CF76IL 46938396 IC50 > 1000 nM T65864 CEQL38 46938397 IC50 > 1000 nM T65864 CW3TD4 46938398 IC50 = 222 nM T65864 CXTM46 46938399 IC50 = 24 nM T65864 CL2K1D 46938400 IC50 = 41 nM T65864 CLW5G8 46938401 IC50 = 50 nM T65864 CAVG61 46938507 IC50 = 72 nM T65864 C7GTV1 46938508 IC50 > 1000 nM T65864 CX47NP 46938509 IC50 = 35 nM T65864 CD58ZL 46938610 IC50 = 110 nM T65864 CKQ5C4 46938612 IC50 = 65 nM T65864 CZM8G3 46938614 IC50 = 259 nM T65864 CD72ZG 46939847 IC50 = 397 nM T65864 CT8F2J 46939848 IC50 = 166 nM T65864 CTB6W4 46943424 IC50 = 3 nM T65864 CJ97YS 49326850 IC50 = 7 nM T65864 C21ZHO 49798293 IC50 = 10000 nM T65864 CNSQ64 49798294 IC50 = 100 nM T65864 C3MLV7 49798295 IC50 = 251.19 nM T65864 CZRY96 49798296 IC50 = 25.12 nM T65864 C0P3OX 49798297 IC50 = 12.59 nM T65864 C9FO3Y 49798328 IC50 = 199.53 nM T65864 CZRY20 49798329 IC50 = 50.12 nM T65864 CA8EX5 49798330 IC50 > 25118.86 nM T65864 C72AUR 49798331 IC50 = 19952.62 nM T65864 CL8R9I 49798332 IC50 = 31.62 nM T65864 C0EF3L 49798352 IC50 = 1258.93 nM T65864 CQ9A4M 49798353 IC50 = 1000 nM T65864 CHSF07 49806372 IC50 > 1000 nM T65864 C9L3XR 49838879 IC50 = 2 nM T65864 CS18HZ 49839481 IC50 > 50000 nM T65864 CF91RS 49843531 IC50 > 10000 nM T65864 C02FRA 49862007 IC50 = 390 nM T65864 CI8HJ9 49862285 IC50 = 2850 nM T65864 CZ4U3X 49862286 IC50 = 176 nM T65864 C47NQS 49862287 IC50 = 287 nM T65864 CV83KC 49862332 IC50 = 68 nM T65864 CXA4U9 49862333 IC50 = 6 nM T65864 CX2BZ1 49862334 IC50 = 441 nM T65864 C01NOJ 49862335 IC50 = 51 nM T65864 CY81LQ 49862397 IC50 = 243 nM T65864 CI0UY7 49862398 IC50 = 18 nM T65864 C71QZD 49862399 IC50 = 168 nM T65864 C3K7MO 49862444 IC50 = 715 nM T65864 CWT04U 49862445 IC50 = 649 nM T65864 CDW5F1 49862446 IC50 = 211 nM T65864 CH07AL 49862447 IC50 = 296 nM T65864 CAP23F 49862493 IC50 = 185 nM T65864 C2MQ7R 49862494 IC50 = 16 nM T65864 CW9Q1F 49862495 IC50 = 231 nM T65864 CWV7G6 49862496 IC50 = 132 nM T65864 C4FQI9 49862557 IC50 = 48.8 nM T65864 C3YZN5 49862558 IC50 = 27.9 nM T65864 CK76ME 49862559 IC50 = 78.2 nM T65864 CBNC06 49862560 IC50 = 393 nM T65864 CTF73G 49862611 IC50 = 39 nM T65864 C4X9TB 49862612 IC50 = 30 nM T65864 CF2GK9 49862613 IC50 = 57 nM T65864 CS2Y7Z 49862614 IC50 = 737 nM T65864 CNA92S 49862661 IC50 = 6 nM T65864 C10NYG 49862707 IC50 = 250 nM T65864 CUS56N 49863686 IC50 = 100000 nM T65864 CIU7C1 49863687 IC50 = 100000 nM T65864 CHL4D9 49863710 IC50 = 100000 nM T65864 CUCO48 49863711 IC50 = 105.5 nM T65864 C83VHI 49864785 IC50 > 100000 nM T65864 C2UTK6 49864850 IC50 > 100000 nM T65864 CAE53W 49865153 IC50 > 100000 nM T65864 C0DRX5 50898538 IC50 = 11000 nM T65864 C09LIX 50899367 IC50 = 9 nM T65864 CQI4A3 50899368 IC50 = 60 nM T65864 C2PH6M 50899468 IC50 = 3 nM T65864 CQ76CZ 50908213 IC50 = 50800 nM T65864 CD2K4R 50908681 Ki > 1000000 nM T65864 C2Y6QS 50938552 IC50 > 10000 nM T65864 CH4FY5 50941455 IC50 > 50000 nM T65864 CBR71Y 50941538 IC50 > 50000 nM T65864 C4BN7W 50941539 IC50 > 50000 nM T65864 C61DVY 50990961 IC50 = 91 nM T65864 CV3UP9 50992247 IC50 = 42 nM T65864 CNWQ30 51035421 IC50 = 135 nM T65864 C9NYP4 51036677 IC50 > 10000 nM T65864 C4WRY3 51037112 IC50 > 10000 nM T65864 CRI28Z 51037948 IC50 > 10000 nM T65864 CQ5XI0 52705183 IC50 = 2390 nM T65864 C8HL1Q 52920793 IC50 > 1000 nM T65864 C95JRW 52920794 IC50 > 1000 nM T65864 C3ZK9J 52920857 IC50 > 1000 nM T65864 CN3D2Y 52936523 IC50 = 158 nM T65864 CHLO87 52936612 IC50 = 223 nM T65864 C23PRQ 52936613 IC50 = 1 nM T65864 CEQN27 52936621 Ki > 1000 nM T65864 CWG75J 52937032 IC50 = 111 nM T65864 CV27AJ 52937134 IC50 = 18 nM T65864 COJ1S5 52937135 IC50 = 20 nM T65864 CU5RP2 52937136 IC50 = 6 nM T65864 CPR7D8 52937239 IC50 = 1 nM T65864 C2JX4E 52937240 IC50 = 12 nM T65864 C78GTF 52937241 IC50 = 7 nM T65864 CRJ5U8 52937242 IC50 = 2 nM T65864 C4TPL6 52937243 IC50 = 1 nM T65864 CI1AW5 52937244 IC50 = 260 nM T65864 C6TW9U 52937346 IC50 = 31 nM T65864 CP1MT0 52940703 IC50 = 19 nM T65864 CTF12V 52940838 IC50 = 1570 nM T65864 C1F0MC 52940949 IC50 = 949 nM T65864 CSTC56 52940962 Ki = 301 nM T65864 C18LMV 52941157 IC50 = 8 nM T65864 CA6BH5 52941226 IC50 > 50000 nM T65864 CMXC68 52941286 IC50 > 50000 nM T65864 CDF2B4 52941332 IC50 = 5 nM T65864 C2BCV1 52941349 Ki = 86 nM T65864 CO5H3E 52941391 Ki = 471 nM T65864 CFIP48 52941393 IC50 = 42 nM T65864 CEO04I 52941436 IC50 = 114 nM T65864 C2A9GP 52941441 Ki = 89 nM T65864 CB7O8A 52941442 Ki = 786 nM T65864 C7F1MP 52941443 Ki = 885 nM T65864 C8KY1N 52941458 IC50 = 4 nM T65864 C7GEY8 52941551 IC50 = 46 nM T65864 CO2NZ4 52941640 IC50 = 52 nM T65864 CJF80K 52941652 Ki = 283 nM T65864 CB32TC 52941869 IC50 = 6280 nM T65864 C78UZD 52941875 IC50 = 6140 nM T65864 C1W8OE 52941889 IC50 = 170 nM T65864 CZ92RI 52941893 IC50 = 38 nM T65864 CJN0P9 52941896 IC50 = 22 nM T65864 C5HU3K 52942035 IC50 = 27 nM T65864 CJ37VI 52942127 IC50 = 160 nM T65864 CEK3W1 52942156 IC50 = 1.6 nM T65864 CU7YS6 52942281 IC50 = 40 nM T65864 C74DCB 52942431 IC50 = 7 nM T65864 CAC3J5 52942507 IC50 > 50000 nM T65864 C3H7ZR 52942530 IC50 = 16 nM T65864 CW5P4Z 52942573 IC50 = 223 nM T65864 CT87PY 52942654 Ki = 157 nM T65864 CRQ67H 52942673 Ki = 291 nM T65864 CV0CZ5 52942728 IC50 = 4 nM T65864 CD5NI0 52942781 IC50 = 573 nM T65864 CYJ53I 52943072 IC50 = 53 nM T65864 C4ZBL5 52943109 IC50 = 27 nM T65864 C26EZU 52943308 IC50 = 280 nM T65864 CB24AN 52943387 Ki = 312 nM T65864 CG3Q6O 52943509 IC50 = 32 nM T65864 C9ZUH4 52943788 IC50 = 2 nM T65864 C03UCH 52943845 Ki = 112 nM T65864 C3Q4RA 52943862 Ki = 1400 nM T65864 CWN1B8 52943885 IC50 = 2 nM T65864 COJF79 52943899 IC50 = 17 nM T65864 CZ4UQ3 52943906 IC50 = 16 nM T65864 CRF45X 52943915 IC50 = 5 nM T65864 CZTM48 52943920 Ki = 1390 nM T65864 CR0EK7 52943970 IC50 = 16 nM T65864 C91VOP 52944103 IC50 = 2.7 nM T65864 CJS85G 52944121 IC50 = 4 nM T65864 CY35NS 52944282 IC50 = 100 nM T65864 CT7MH1 52944298 IC50 = 90 nM T65864 C26CXH 52944302 IC50 = 180 nM T65864 CXN1V4 52944905 IC50 = 8 nM T65864 CB1UJ7 52944909 IC50 > 50000 nM T65864 CQPI17 52944927 IC50 = 7 nM T65864 CYO3A9 52945030 IC50 = 2 nM T65864 CSZ98U 52945031 IC50 = 2 nM T65864 CIL7G6 52945080 Ki = 140 nM T65864 C4AC8V 52945117 Ki = 735 nM T65864 CY15LQ 52945517 IC50 = 2260 nM T65864 C2HT3O 52945518 IC50 = 18 nM T65864 CDT78K 52945802 IC50 = 3.9 nM T65864 C5LVU9 52945951 IC50 = 770 nM T65864 C50FTK 52945955 IC50 = 10 nM T65864 CCMX82 52946092 IC50 > 50000 nM T65864 CJ25IG 52946108 IC50 = 14 nM T65864 C4PT7O 52946291 Ki = 336 nM T65864 C0BC5R 52946292 Ki > 3900 nM T65864 CMK9Q5 52946354 IC50 = 6 nM T65864 C18HZC 52946366 Ki > 3900 nM T65864 C1XOR6 52946367 IC50 = 8 nM T65864 C7WZ4T 52946477 IC50 = 1200 nM T65864 C1Z6NM 52946501 IC50 = 130 nM T65864 C13QHL 52946670 IC50 > 10000 nM T65864 C5CED2 52946709 IC50 = 790 nM T65864 C6PV4R 52946727 IC50 = 490 nM T65864 C2LTU3 52946735 IC50 = 100 nM T65864 CDYR79 52946741 IC50 = 170 nM T65864 CC8W4I 52946743 IC50 = 280 nM T65864 CKB5J2 52946752 IC50 = 130 nM T65864 CMOF71 52946757 IC50 = 140 nM T65864 C9C8WO 52946761 IC50 = 440 nM T65864 CBW9V7 52946875 IC50 = 180 nM T65864 CI91LF 52946884 IC50 = 2240 nM T65864 CMF42A 52946979 IC50 = 320 nM T65864 CHFY62 52946980 IC50 = 100 nM T65864 C0KCQ3 52947055 IC50 = 314 nM T65864 C3YW2A 52947365 IC50 = 6 nM T65864 CZY80A 52947401 IC50 > 1000 nM T65864 C1M9DQ 52947439 IC50 = 22 nM T65864 C3DTS8 52947470 IC50 = 859 nM T65864 CJ4Q3P 52947527 Ki = 433 nM T65864 C9C7OT 52947528 Ki = 1450 nM T65864 CBX2M5 52947595 IC50 = 5 nM T65864 CF67LA 52947611 IC50 = 2.1 nM T65864 CP8AX1 52947723 IC50 = 780 nM T65864 CA6XF0 52947931 IC50 = 400 nM T65864 C96UGN 52947932 IC50 = 160 nM T65864 CON8L1 52947941 IC50 = 13 nM T65864 C78QUA 52947960 IC50 = 1490 nM T65864 C7HWY0 52947961 IC50 = 93 nM T65864 C47CRW 52947977 IC50 = 75 nM T65864 CN0J1O 52948100 IC50 = 225 nM T65864 CU5OA3 52948191 Ki = 327 nM T65864 CN0KA4 52948220 IC50 = 3.1 nM T65864 C31KRC 52948227 IC50 = 2.9 nM T65864 CB87ZN 52948381 IC50 = 150 nM T65864 CLU92X 52948565 IC50 > 50000 nM T65864 CDXL70 52948593 IC50 > 50000 nM T65864 C9FV8O 52948677 IC50 = 3 nM T65864 CS7Q4W 52948733 Ki = 715 nM T65864 CXOQ20 52948737 IC50 = 3940 nM T65864 C9Z2RY 52948828 IC50 = 5 nM T65864 C8M1HJ 52948905 IC50 = 240 nM T65864 CI9XF2 52948960 IC50 = 570 nM T65864 CTC18Q 52948967 IC50 = 520 nM T65864 CZ6MS5 52949170 IC50 = 27 nM T65864 C7F2SW 52949171 IC50 = 180 nM T65864 CYUW97 52949194 IC50 = 150 nM T65864 C1UM7B 52949201 IC50 = 17 nM T65864 CWAV65 52949209 IC50 = 330 nM T65864 C26AXT 52949261 Ki = 176 nM T65864 C01XZI 52949301 Ki = 252 nM T65864 CNB2J0 52949346 IC50 > 1000 nM T65864 C8IV2N 52949429 IC50 = 14 nM T65864 CW3G8L 52949622 IC50 = 1620 nM T65864 C65ZXV 52949623 IC50 = 170 nM T65864 CBG3Q0 52949627 IC50 = 1140 nM T65864 CIVE91 52949671 IC50 = 5 nM T65864 C6TG2B 52949802 IC50 = 2 nM T65864 CMT75N 52949817 IC50 > 50000 nM T65864 CR9JT3 52949868 IC50 = 52 nM T65864 C0V7QF 52949942 Ki > 3900 nM T65864 CS7R1C 52949978 IC50 = 17 nM T65864 CJN69P 52950128 IC50 = 7 nM T65864 C6EM7B 53237688 IC50 = 2 nM T65864 C6KS3N 53237689 IC50 = 12 nM T65864 CE28GW 53237690 IC50 = 120 nM T65864 CHG40F 53237691 IC50 = 26 nM T65864 C8RE9F 53237692 IC50 = 180 nM T65864 CKU14E 53237693 IC50 = 37 nM T65864 CJ9PC2 53237915 IC50 = 2 nM T65864 CE8SK3 53237916 IC50 = 1080 nM T65864 CSG8A7 53237917 IC50 = 12 nM T65864 CI14NP 53237918 IC50 = 3 nM T65864 CV0QM5 53237919 IC50 = 69 nM T65864 CE82FQ 53237920 IC50 = 207 nM T65864 CT2YZ1 53238147 IC50 = 95 nM T65864 C34QDW 53238148 IC50 = 34 nM T65864 CG6I2V 53238149 IC50 = 17 nM T65864 C01KZJ 53238150 IC50 = 1340 nM T65864 C2X4DU 53238151 IC50 = 403 nM T65864 CDQ4V0 53238152 IC50 = 1265 nM T65864 CH51WL 53238153 IC50 = 840 nM T65864 C17FWR 53238381 IC50 = 21 nM T65864 CY38TE 53238382 IC50 = 34 nM T65864 C3X7EU 53238383 IC50 = 6 nM T65864 CNW52E 53238384 IC50 = 141 nM T65864 CWV8N3 53238385 IC50 = 200 nM T65864 C3C0IR 53238386 IC50 = 45 nM T65864 CG36MF 53238608 IC50 = 50 nM T65864 C37PYI 53238609 IC50 = 27 nM T65864 C0ZO9T 53238610 IC50 = 36 nM T65864 CK35NW 53238611 IC50 = 197 nM T65864 CV0AQ9 53238836 IC50 = 129 nM T65864 CTU7F6 53238837 IC50 = 12 nM T65864 C8IOE2 53238838 IC50 = 11 nM T65864 COX81P 53238839 IC50 = 11 nM T65864 CCMV80 53238840 IC50 = 450 nM T65864 COZ1Y3 53238841 IC50 = 77 nM T65864 C85SHV 53239057 IC50 = 168 nM T65864 CI74SF 53239058 IC50 = 25 nM T65864 CSNK01 53239059 IC50 = 29 nM T65864 CHJZ49 53239060 IC50 = 19 nM T65864 C90HFT 53239061 IC50 = 31 nM T65864 CN9X0C 53239062 IC50 = 161 nM T65864 CZR50O 53239984 IC50 = 151 nM T65864 C9RX3G 53239985 IC50 = 134 nM T65864 C6DC4S 53241447 IC50 = 8 nM T65864 CBTX53 53317412 IC50 > 50000 nM T65864 COCN94 53317413 IC50 > 50000 nM T65864 CHC29T 53317414 IC50 > 50000 nM T65864 C82LCE 53317415 IC50 > 50000 nM T65864 CR0DJ1 53317416 IC50 > 50000 nM T65864 CP7T3N 53318709 IC50 > 50000 nM T65864 C3TAC2 53320021 IC50 > 5000 nM T65864 COPI53 53321333 IC50 > 50000 nM T65864 C0GLS5 53321334 IC50 > 50000 nM T65864 C2V0QU 53321577 IC50 > 50000 nM T65864 COG9J2 53322644 IC50 > 50000 nM T65864 CUR1A6 53322645 IC50 > 50000 nM T65864 C9SHJ0 53323985 IC50 > 50000 nM T65864 C49MDG 53323986 IC50 > 50000 nM T65864 C3AVG0 53323987 IC50 > 50000 nM T65864 C38RXW 53323989 IC50 > 50000 nM T65864 C2W9OA 53324451 IC50 > 10000 nM T65864 C8VPW5 53325283 IC50 > 50000 nM T65864 CA3X2Q 53325284 IC50 > 50000 nM T65864 CIG7X9 53325285 IC50 > 50000 nM T65864 C4A8JK 53325286 IC50 > 50000 nM T65864 CNT50E 53325288 IC50 > 50000 nM T65864 CV7I4O 53326555 IC50 > 50000 nM T65864 C27IBZ 53326556 IC50 > 50000 nM T65864 C5UK3J 53326557 IC50 > 50000 nM T65864 CVJ6K9 53326558 IC50 > 50000 nM T65864 C8NA4L 53384644 IC50 = 22 nM T65864 CP1FH5 53391990 IC50 = 2 nM T65864 C3ANK0 53470402 IC50 = 3641 nM T65864 C4JCT1 53476174 IC50 = 11 nM T65864 C0U2OR 54578934 IC50 > 1000 nM T65864 CDZ09I 54578935 IC50 > 1000 nM T65864 CI6UG7 54578936 IC50 > 1000 nM T65864 C0WM1Y 54580506 IC50 > 1000 nM T65864 C4W7BZ 54580507 IC50 > 1000 nM T65864 C2AUV0 54580508 IC50 > 1000 nM T65864 CF9HP7 54580509 IC50 > 1000 nM T65864 C6MXZ8 54580510 IC50 > 1000 nM T65864 CCVR53 54580511 IC50 = 630 nM T65864 C5CKG1 54580689 IC50 = 45 nM T65864 C8TH5W 54580690 IC50 = 2200 nM T65864 C0V7UY 54580691 IC50 = 10400 nM T65864 C8L0PY 54581453 IC50 = 85.11 nM T65864 CEP04I 54581525 IC50 > 1000 nM T65864 CCM64U 54581691 IC50 = 1000 nM T65864 CZO9H1 54581692 IC50 = 420 nM T65864 CEV07C 54581693 IC50 = 38 nM T65864 C5V6OY 54582175 IC50 > 30000 nM T65864 CU30TM 54582521 IC50 > 1000 nM T65864 COT7C9 54583645 IC50 = 59 nM T65864 C6SV3D 54584455 IC50 = 453 nM T65864 CKAX21 54584471 IC50 > 1000 nM T65864 CK73XV 54584619 IC50 = 3580 nM T65864 CBJ01K 54584630 IC50 = 690 nM T65864 C0NC9L 54585425 IC50 > 1000 nM T65864 CB6XT7 54585426 IC50 > 1000 nM T65864 CC84VU 54585567 IC50 = 84 nM T65864 CNUP53 54586040 IC50 = 4700 nM T65864 CA6L5Q 54586370 IC50 = 316.23 nM T65864 CA4GI9 54586383 IC50 > 1000 nM T65864 C6VFC4 54586384 IC50 > 1000 nM T65864 C5MZ2T 54586385 IC50 > 1000 nM T65864 CIL4A3 54586547 IC50 = 257 nM T65864 CIUC72 54587577 IC50 = 100 nM T65864 COW9Z6 54587582 IC50 = 795 nM T65864 C9UG6V 54587823 IC50 = 230 nM T65864 C3EJ0P 54673693 IC50 > 5000 nM T65864 CET93B 54673697 IC50 > 5000 nM T65864 CE1ZK6 54759168 IC50 > 10000 nM T65864 C1XS2J 54760383 IC50 = 230 nM T65864 C3HTE0 54765510 IC50 = 2420 nM T65864 CCZ2V9 54765512 IC50 = 533 nM T65864 C9M0SO 54765514 IC50 = 844 nM T65864 CS0HQ8 54765517 IC50 = 2230 nM T65864 CSNW70 54765683 IC50 = 384 nM T65864 C6FDL2 54766012 IC50 = 2290 nM T65864 C15TGK 54766018 IC50 = 4890 nM T65864 C3MJ8Y 54766164 IC50 = 820 nM T65864 C7AY9N 54766165 IC50 = 3930 nM T65864 CLKF74 54766166 IC50 = 2540 nM T65864 CH3V8A 54766167 IC50 = 1250 nM T65864 C6HX3D 54766168 IC50 = 500 nM T65864 C9E4LP 54766169 IC50 > 10000 nM T65864 CL75WK 54766171 IC50 = 6240 nM T65864 CD36HW 54766320 IC50 = 730 nM T65864 CL71CV 54766321 IC50 = 8640 nM T65864 CG4L7Y 54766322 IC50 = 9300 nM T65864 CA74KU 54766323 IC50 = 3890 nM T65864 C25FDK 54766324 IC50 = 1070 nM T65864 C21KGR 54766325 IC50 = 1980 nM T65864 CM92AB 54766465 IC50 = 870 nM T65864 C64JAV 54766466 IC50 > 10000 nM T65864 CEX96A 54766467 IC50 = 1940 nM T65864 CVG4X7 54766468 IC50 = 1310 nM T65864 C78SKD 54766469 IC50 > 10000 nM T65864 CWV13U 54766470 IC50 = 3490 nM T65864 CV9JN8 54766620 IC50 > 10000 nM T65864 C5SK9R 54766621 IC50 = 3000 nM T65864 CG1B5U 54766622 IC50 = 1530 nM T65864 C7REA0 54766623 IC50 = 1180 nM T65864 C65HJI 54766624 IC50 = 1100 nM T65864 CD96AG 54766625 IC50 = 1210 nM T65864 CT51IV 54766773 IC50 > 10000 nM T65864 C2DIH5 54766774 IC50 = 2050 nM T65864 C9W1SM 54766775 IC50 = 1460 nM T65864 C56PNG 54766776 IC50 > 10000 nM T65864 CJO9Y0 54766778 IC50 = 3680 nM T65864 CUJ2A9 54766930 IC50 = 2430 nM T65864 C7YO8F 54766931 IC50 > 10000 nM T65864 C8OXL1 54766932 IC50 > 10000 nM T65864 CZ5JR9 54766933 IC50 > 10000 nM T65864 C7R6PT 54766934 IC50 = 2850 nM T65864 C2GO1J 54767085 IC50 = 2560 nM T65864 CCYX42 54767086 IC50 = 1860 nM T65864 C41UWF 54767087 IC50 > 10000 nM T65864 C1E2PB 54767088 IC50 = 1300 nM T65864 CFB9S3 54767243 IC50 = 700 nM T65864 CUV96X 54767245 IC50 > 10000 nM T65864 C7K5SJ 54767246 IC50 = 3640 nM T65864 CW0GJ7 54767248 IC50 = 1500 nM T65864 CN9YX4 54767249 IC50 = 3940 nM T65864 CG6RC9 54767416 IC50 > 10000 nM T65864 C92THY 54767417 IC50 = 1280 nM T65864 CP84QJ 54767418 IC50 = 1390 nM T65864 CQY04U 54767419 IC50 = 1630 nM T65864 CFZ97I 54767420 IC50 = 2830 nM T65864 CXO65G 54767583 IC50 = 178 nM T65864 CPG8U6 54767584 IC50 = 393 nM T65864 C5T1ZU 54767753 IC50 = 2480 nM T65864 CS06AD 54767754 IC50 = 4110 nM T65864 C3E0RV 54767755 IC50 = 4100 nM T65864 CFL9P5 54767911 IC50 = 1710 nM T65864 CV4I2C 54767912 IC50 = 259 nM T65864 CPW58S 54769997 IC50 > 1000 nM T65864 CLR3Y9 54769998 IC50 > 1000 nM T65864 C1O3UI 54770205 IC50 > 1000 nM T65864 CL6FY2 54770206 IC50 > 1000 nM T65864 CD6R9I 54770207 IC50 > 1000 nM T65864 C2ZV0I 54770208 IC50 > 1000 nM T65864 CN4H9Z 54770209 IC50 > 1000 nM T65864 CXH87U 54770427 IC50 > 1000 nM T65864 C29OBP 54770428 IC50 > 1000 nM T65864 CZ38LT 54770429 IC50 > 1000 nM T65864 C12POE 54770430 IC50 > 1000 nM T65864 CSW69T 54770431 IC50 > 1000 nM T65864 C8VW1G 54770641 IC50 > 1000 nM T65864 C4U7BS 54771536 IC50 = 142 nM T65864 CS1R4P 54771537 IC50 > 10000 nM T65864 C7G2HI 54771538 IC50 = 7810 nM T65864 CG7X5S 54771759 IC50 = 1540 nM T65864 CGSX68 54771760 IC50 > 10000 nM T65864 C9C4VJ 54771761 IC50 > 10000 nM T65864 CT8E3Q 54771762 IC50 = 1410 nM T65864 C70GUO 54771763 IC50 > 10000 nM T65864 CL48YQ 54771764 IC50 = 3980 nM T65864 CKA4M2 55786207 IC50 = 8 nM T65864 CQM45J 56589562 IC50 = 34 nM T65864 C91JFI 56589563 IC50 = 17 nM T65864 C0D1CP 56594665 IC50 = 813 nM T65864 C7H8CT 56594666 IC50 = 1380 nM T65864 CNQ1O5 56594667 IC50 = 21 nM T65864 CZJ72C 56594668 IC50 = 39 nM T65864 C8BOP5 56594669 IC50 = 761 nM T65864 C3AH4G 56594670 IC50 = 45 nM T65864 C1U4JW 56594794 IC50 = 35 nM T65864 CM8JX1 56604907 IC50 = 1000 nM T65864 CS68PK 56659526 IC50 = 38 nM T65864 CK3CF4 56659737 IC50 = 5 nM T65864 C2SNV0 56659738 IC50 = 55 nM T65864 CE1O3B 56661803 IC50 > 50000 nM T65864 CGD72U 56662990 IC50 = 3 nM T65864 C45WTE 56663206 IC50 = 27 nM T65864 C6TM5W 56663207 IC50 = 230 nM T65864 CS0VX8 56663208 IC50 = 55 nM T65864 C84KVY 56663285 IC50 = 12 nM T65864 CY1PA8 56663286 IC50 = 59 nM T65864 CY3MQ8 56663287 IC50 = 36 nM T65864 CHJX02 56666448 IC50 = 6 nM T65864 CXF2T5 56666645 IC50 = 19 nM T65864 C26CKY 56666646 IC50 = 12 nM T65864 CJKH04 56666649 IC50 = 15 nM T65864 CT2P7H 56670061 IC50 = 44 nM T65864 C9R3KY 56670062 IC50 = 11 nM T65864 C29ZDN 56670138 IC50 = 140 nM T65864 C3WYD7 56670139 IC50 = 35 nM T65864 CB64JZ 56673341 IC50 = 2 nM T65864 CLGU31 56673356 IC50 = 27 nM T65864 C5C9OE 56673357 IC50 = 12 nM T65864 C0AKO6 56673497 IC50 = 15 nM T65864 CV60YB 56673498 IC50 = 142 nM T65864 CADI17 56673550 Ki = 290 nM T65864 CC2L3G 56673581 IC50 = 88 nM T65864 CWHN47 56673582 IC50 = 240 nM T65864 CX76JT 56673586 IC50 = 10 nM T65864 C1E8IX 56676901 IC50 = 6 nM T65864 CKVS08 56676902 IC50 = 45 nM T65864 CGC41K 56676903 IC50 > 1000 nM T65864 C65ECF 56676912 IC50 = 52 nM T65864 C5XY9H 56680004 IC50 = 193 nM T65864 C9BH3M 56680220 IC50 = 18 nM T65864 CDHO64 56680302 IC50 = 19 nM T65864 C9DO8G 56682210 IC50 > 50000 nM T65864 C04IWS 56683552 IC50 = 3 nM T65864 CZH58B 56683561 IC50 = 10 nM T65864 C2PQ4W 56683623 IC50 = 14 nM T65864 CT4E8R 56832546 IC50 > 100000 nM T65864 CJ4LC1 56834581 IC50 > 1000 nM T65864 C2C3NH 56834583 IC50 = 422 nM T65864 CRT7P9 56834584 IC50 = 1400 nM T65864 CU2JR7 56834585 IC50 = 81 nM T65864 CH1V3X 56834671 IC50 = 37 nM T65864 CN45UL 56834672 IC50 = 29 nM T65864 CN97QM 56834673 IC50 = 14 nM T65864 C3OE9X 56834674 IC50 = 17 nM T65864 CG3P9V 56834675 IC50 = 11 nM T65864 CFY4X0 56834676 IC50 = 0.26 nM T65864 C1NQ7A 56834762 IC50 = 0.13 nM T65864 CW1U0X 56834763 IC50 = 0.5 nM T65864 CIE7J3 56834764 IC50 = 0.46 nM T65864 CB5Z1I 56834765 IC50 = 9 nM T65864 CTO6N5 56834943 IC50 = 220 nM T65864 C5LJE8 56951456 IC50 = 1.1 nM T65864 C6N0ZI 56951457 IC50 = 4.9 nM T65864 CL90EM 56951458 IC50 = 1.2 nM T65864 CG63ZF 56962313 IC50 = 9 nM T65864 CJ47MX 56963907 IC50 > 10000 nM T65864 C9L6FD 56963908 IC50 > 10000 nM T65864 CE50IB 56963909 IC50 > 10000 nM T65864 CJZH10 57328694 IC50 = 639 nM T65864 CDP45J 57390517 IC50 = 1300 nM T65864 C28LIB 57390518 IC50 = 3500 nM T65864 C8DZ1N 57390519 IC50 = 510 nM T65864 C7K4LJ 57390520 IC50 = 210 nM T65864 CP7Z1K 57390703 IC50 = 2 nM T65864 CT4KZ6 57390882 IC50 = 4.1 nM T65864 CDW10R 57390883 IC50 = 1.6 nM T65864 CHU75J 57390951 IC50 > 3000 nM T65864 CG51FX 57392289 IC50 = 210 nM T65864 C62EJX 57392507 IC50 = 14 nM T65864 C9E0BK 57392508 IC50 = 31 nM T65864 CBD87K 57392509 IC50 = 19 nM T65864 CL18AV 57392510 IC50 = 39 nM T65864 C17PSI 57392650 IC50 = 1 nM T65864 CSYJ61 57392738 IC50 = 910 nM T65864 C2IZ3W 57392739 IC50 = 4200 nM T65864 C3I2UA 57392752 IC50 = 87 nM T65864 CJHS69 57392857 IC50 = 34 nM T65864 C9P1SC 57393560 IC50 = 490 nM T65864 CVH4X0 57394043 IC50 = 1600 nM T65864 CD05MZ 57394214 IC50 = 13 nM T65864 CHAC45 57394395 IC50 = 1.3 nM T65864 C52RAH 57394396 IC50 = 2 nM T65864 CDW16B 57394397 IC50 = 6.3 nM T65864 CIYF92 57394398 IC50 = 1 nM T65864 C03CNR 57394466 IC50 = 560 nM T65864 CX9B4S 57394467 IC50 = 290 nM T65864 C1EYU6 57394468 IC50 > 3000 nM T65864 CV9W8C 57395293 IC50 = 240 nM T65864 CQ2A1B 57395802 IC50 = 2800 nM T65864 CDE3T9 57395979 IC50 = 80 nM T65864 CW7XA9 57397040 IC50 = 490 nM T65864 CU4FW8 57397383 IC50 = 7.6 nM T65864 C4V9RN 57398023 IC50 = 160 nM T65864 CZI7A2 57398024 IC50 = 6400 nM T65864 C4RJ0E 57398025 IC50 > 3000 nM T65864 CY12SA 57398677 IC50 = 2.8 nM T65864 CDUS89 57399441 IC50 = 13 nM T65864 CZY93W 57399442 IC50 = 29 nM T65864 CPCF09 57399443 IC50 = 73 nM T65864 C2CIY0 57399621 IC50 = 1.4 nM T65864 CX9ZR3 57399622 IC50 = 16.9 nM T65864 CE76QR 57399681 IC50 = 6200 nM T65864 CRNJ52 57399682 IC50 = 860 nM T65864 CIH8D6 57399817 IC50 = 90 nM T65864 C2O3ZP 57400111 Ki = 14 nM T65864 CLI72R 57401441 IC50 = 2700 nM T65864 CC7N3H 57401442 IC50 = 230 nM T65864 CPY13U 57401443 IC50 > 3000 nM T65864 C8FQH3 57402785 IC50 > 30000 nM T65864 C4LK0M 57402955 IC50 = 140 nM T65864 C2YZ7E 57403132 IC50 = 1.9 nM T65864 CKE0V9 57403185 IC50 = 980 nM T65864 CAC91M 57467724 IC50 = 45.6 nM T65864 C6UAN1 57467725 IC50 = 792 nM T65864 CE59QS 57505507 IC50 > 1000 nM T65864 C4K8HW 57834331 IC50 = 14 nM T65864 C5WX1O 57834340 IC50 = 22 nM T65864 C3CL2Y 57834396 IC50 = 19 nM T65864 CVK0G4 58056356 IC50 > 50000 nM T65864 C6VQ8S 58328161 IC50 = 23 nM T65864 CYZ6X2 58328191 IC50 = 35 nM T65864 C7WX9H 58328291 IC50 = 32 nM T65864 C2JW1C 58328294 IC50 = 34 nM T65864 C6HR5F 58416745 IC50 = 60 nM T65864 CRY9K7 58416748 IC50 = 11 nM T65864 CYI32L 58532548 IC50 = 38 nM T65864 CKXE59 58577987 IC50 = 2350 nM T65864 CBNJ31 58577988 IC50 = 2270 nM T65864 CY7WR0 58577989 IC50 = 699 nM T65864 CAN79D 58577996 IC50 = 422 nM T65864 CTX23R 58577998 IC50 > 10000 nM T65864 C3PC5S 58608697 IC50 = 1.86 nM T65864 CL7G8Y 58659496 IC50 = 105 nM T65864 CF4S6Q 58688403 IC50 = 590 nM T65864 CVO46Z 58688633 IC50 = 1999 nM T65864 CG4ID2 59151856 IC50 = 35 nM T65864 CQL8H7 59151869 IC50 = 3 nM T65864 CZ5S1G 59151878 IC50 = 13 nM T65864 CDTW26 59151884 IC50 = 14 nM T65864 C9AOP6 59151928 IC50 = 4 nM T65864 CL57UP 59151937 IC50 = 11 nM T65864 COMG36 59151943 IC50 = 1500 nM T65864 C8GEJ7 59151971 IC50 = 5 nM T65864 CXJ63M 59603829 IC50 = 36000 nM T65864 CQEU96 59603842 IC50 = 1400 nM T65864 C8MS1C 59749702 IC50 = 4 nM T65864 CIGB91 59759551 IC50 = 73 nM T65864 C28ZVH 59759556 IC50 = 23 nM T65864 CU6CX0 59759575 IC50 = 84 nM T65864 CT07VZ 59759607 IC50 = 9.4 nM T65864 CIO5W6 59759608 IC50 = 34 nM T65864 CJXO41 59759622 IC50 = 23 nM T65864 CLM62Y 59759659 IC50 = 11 nM T65864 C3UAB6 59759685 IC50 = 290 nM T65864 CNGL17 59759724 IC50 = 56 nM T65864 CL92GP 59761390 IC50 = 46 nM T65864 CH21LA 59761399 IC50 = 13 nM T65864 C5GAK1 59761424 IC50 = 5.4 nM T65864 C6DNV0 59761433 IC50 = 7.7 nM T65864 CYV4E3 59761440 IC50 = 14 nM T65864 CIO25V 59761450 IC50 = 11 nM T65864 CFSO82 59761454 IC50 = 41 nM T65864 CIM3Z0 59761458 IC50 = 8.6 nM T65864 C3MJC9 59761459 IC50 = 4.1 nM T65864 CRJ54F 59761462 IC50 = 4.1 nM T65864 CT51GX 59761498 IC50 = 8.9 nM T65864 CS41QF 59761509 IC50 = 3.8 nM T65864 CI3VU5 59761513 IC50 = 3.8 nM T65864 C6X0WG 60034040 IC50 = 24 nM T65864 C1MR8Q 60097495 IC50 > 5000 nM T65864 CKT2R0 60148471 IC50 = 1500 nM T65864 CWV37N 60166859 IC50 = 70 nM T65864 CT1IG2 60166860 IC50 = 50 nM T65864 CZ65BW 60166861 IC50 = 3530 nM T65864 CT0K6L 60166862 IC50 = 30 nM T65864 CY4P8L 60166863 IC50 = 60 nM T65864 C83GRK 60166864 IC50 = 60 nM T65864 CSJ9O8 60166988 IC50 = 40 nM T65864 C4UY3Q 60166989 IC50 = 10 nM T65864 C6RE9C 60166990 IC50 = 10 nM T65864 C9DWE0 60166991 IC50 = 8 nM T65864 C6LW5J 60166992 IC50 = 100 nM T65864 CVC7P2 60167137 IC50 = 20 nM T65864 C0UG7S 60167138 IC50 = 20 nM T65864 CJ2UL8 60167139 IC50 = 30 nM T65864 CT7S3V 60167140 IC50 = 360 nM T65864 CE4P6J 60167141 IC50 = 5200 nM T65864 CO26NI 60167281 IC50 = 70 nM T65864 CYJS51 62705677 IC50 = 13 nM T65864 CE7Q3S 66557865 IC50 = 35 nM T65864 C38AHD 66632799 IC50 > 10000 nM T65864 C1HSE0 67035086 IC50 = 4800 nM T65864 CWI6K5 67035106 IC50 > 10000 nM T65864 C38RGB 67035556 IC50 > 10000 nM T65864 C26TWY 67148905 IC50 = 5 nM T65864 C71VZT 67196472 IC50 = 141 nM T65864 C5PT8D 67197758 IC50 = 33.2 nM T65864 CJ4T0Y 67198791 IC50 = 294 nM T65864 CSWF87 67198998 IC50 = 1010 nM T65864 CM45QD 67199939 IC50 = 8.43 nM T65864 CV63UL 67240318 IC50 > 10000 nM T65864 C32LFE 67374618 IC50 = 15000 nM T65864 C46VLA 67374621 IC50 = 5900 nM T65864 CLKN38 67375395 IC50 = 15000 nM T65864 C5BFR4 67378301 IC50 = 3500 nM T65864 CKB37H 67379186 IC50 = 1600 nM T65864 C8M9VH 67379418 IC50 = 14000 nM T65864 CNT0W7 67468470 IC50 > 5000 nM T65864 CLD91A 67468733 IC50 > 5000 nM T65864 C3U7GQ 67469028 IC50 > 5000 nM T65864 CZC9M5 67469084 IC50 = 5119 nM T65864 C8I7GC 68293638 IC50 > 10000 nM T65864 CD56XK 68293660 IC50 > 10000 nM T65864 CAWC35 68621678 IC50 > 1000 nM T65864 C07NTU 68747277 IC50 = 30000 nM T65864 CD9J0Y 68778068 IC50 = 30000 nM T65864 CG16HX 68780878 IC50 = 36000 nM T65864 C5DGR9 69036886 IC50 = 10000 nM T65864 CUI37S 69227465 IC50 = 108 nM T65864 CKJT70 69692723 IC50 = 5.72 nM T65864 C3GTU1 69762142 IC50 > 10000 nM T65864 C64BAZ 70678406 IC50 = 1 nM T65864 CQ0NH3 70681601 IC50 = 708 nM T65864 CMH9R7 70681602 IC50 = 730 nM T65864 CE73DF 70681603 IC50 > 2200 nM T65864 CX0UK8 70681617 IC50 = 199.53 nM T65864 CMGA79 70682196 IC50 = 100000 nM T65864 C4HN7F 70682754 IC50 = 5530 nM T65864 CGK6B1 70682755 IC50 = 3780 nM T65864 C0V7PS 70682756 IC50 = 5860 nM T65864 C6SDX9 70682757 IC50 > 10000 nM T65864 CGCP65 70682763 IC50 > 10000 nM T65864 CS7F5Y 70683717 IC50 = 81.28 nM T65864 CH0T3O 70684298 IC50 = 19000 nM T65864 C4DKI7 70684836 IC50 = 5370 nM T65864 CV37TR 70684847 IC50 > 10000 nM T65864 CFS6H3 70684848 IC50 = 6190 nM T65864 CKC26J 70685673 IC50 = 2100 nM T65864 C9A6KW 70685867 IC50 = 64.57 nM T65864 C8GQ6X 70685868 IC50 = 16.6 nM T65864 CGO1T3 70685869 IC50 = 346.74 nM T65864 C82FIP 70686752 IC50 > 10000 nM T65864 CMA38X 70686991 IC50 > 10000 nM T65864 C87LYT 70686992 IC50 > 10000 nM T65864 CXJ76O 70687994 IC50 = 15 nM T65864 C6X4EB 70687995 IC50 = 20 nM T65864 CP4K6M 70687996 IC50 = 4168.69 nM T65864 CJ30DE 70687997 IC50 = 155 nM T65864 COX8Z2 70687998 IC50 = 525 nM T65864 CTCF71 70688555 IC50 = 12000 nM T65864 C0QX3Y 70688829 IC50 > 10000 nM T65864 C8N7IV 70689057 IC50 = 3280 nM T65864 CX2Y5O 70689058 IC50 = 7390 nM T65864 CTH0A9 70689059 IC50 > 10000 nM T65864 C0BIE1 70689068 IC50 > 10000 nM T65864 C8PC1T 70689069 IC50 = 7990 nM T65864 C0IC3J 70689070 IC50 > 10000 nM T65864 C1DVU0 70689071 IC50 > 10000 nM T65864 C8BJ6C 70690017 IC50 = 220 nM T65864 CYEZ06 70690018 IC50 = 1949.84 nM T65864 CU1CM2 70690019 IC50 = 14 nM T65864 CB1A6I 70690020 IC50 = 107.15 nM T65864 C08WPT 70690038 IC50 = 261 nM T65864 CNER46 70690618 IC50 = 100000 nM T65864 CQ8HE2 70690944 IC50 > 30000 nM T65864 CJL0N2 70691169 IC50 > 10000 nM T65864 CN25KI 70691183 IC50 > 10000 nM T65864 C8X6QU 70691184 IC50 > 10000 nM T65864 C78SZC 70692177 IC50 = 20.42 nM T65864 CZ7GQ9 70692192 IC50 = 1288.25 nM T65864 CTYA67 70692760 IC50 = 100000 nM T65864 CSOT12 70693058 IC50 > 10000 nM T65864 CS6NW3 70693059 IC50 > 10000 nM T65864 CJD7K6 70693280 IC50 > 10000 nM T65864 CC0W1O 70693281 IC50 > 10000 nM T65864 C2SUY0 70694238 IC50 = 1200 nM T65864 CU9Q7G 70694239 IC50 = 181 nM T65864 CBI12T 70694240 IC50 = 1535 nM T65864 C8SLN0 70694241 IC50 > 50118.72 nM T65864 C45SUB 70694800 IC50 = 15000 nM T65864 C95IBJ 70694801 IC50 = 22000 nM T65864 C13FWG 70695135 IC50 > 30000 nM T65864 C7ZT3R 70695370 IC50 = 3530 nM T65864 CY8SW6 70695371 IC50 > 10000 nM T65864 CSUD72 70695372 IC50 = 3820 nM T65864 CQH26P 70696332 IC50 = 89.13 nM T65864 CD09ZQ 70696333 IC50 = 1258.93 nM T65864 CGM7X8 70696348 IC50 = 1445.44 nM T65864 C2SWX1 70696850 IC50 = 100000 nM T65864 C0VZB2 70697173 IC50 > 30000 nM T65864 C9SU2M 70697187 IC50 = 3940 nM T65864 CAQY83 70697381 IC50 > 10000 nM T65864 C0I8GU 70697382 IC50 = 9200 nM T65864 CYW19K 70697383 IC50 > 10000 nM T65864 C91VYF 70697384 IC50 = 7200 nM T65864 C7HS8G 70697385 IC50 = 3580 nM T65864 C3GH1P 70697386 IC50 > 10000 nM T65864 C3W5GQ 70697400 IC50 > 10000 nM T65864 CKH76B 70697401 IC50 = 8820 nM T65864 CR2U5G 70697402 IC50 > 10000 nM T65864 C0N7DY 71449477 IC50 = 290 nM T65864 CG1LX5 71449963 IC50 = 130 nM T65864 C79EGP 71449964 IC50 = 4800 nM T65864 C27ATO 71449965 IC50 = 5 nM T65864 C4P1GW 71449966 IC50 = 17 nM T65864 CWY94O 71450102 IC50 = 39 nM T65864 CSZ70A 71450103 IC50 = 8 nM T65864 C8BF9M 71450324 IC50 = 4300 nM T65864 CEO6L0 71450325 IC50 = 32 nM T65864 CV4XQ7 71450326 IC50 = 20 nM T65864 C92XIV 71450327 IC50 = 100 nM T65864 CA4FZ9 71450328 IC50 = 350 nM T65864 C69SEG 71450329 IC50 = 300 nM T65864 CR1Y0O 71450330 IC50 = 2700 nM T65864 C3JD0U 71450331 IC50 = 160 nM T65864 C1FMW5 71451789 IC50 = 37 nM T65864 C2TGF7 71451790 IC50 = 20 nM T65864 CCPA08 71451911 IC50 = 70 nM T65864 C58BSC 71451912 IC50 = 108 nM T65864 C24WSE 71451913 IC50 = 451 nM T65864 CML3C4 71451914 IC50 = 153 nM T65864 C4EK3L 71452132 IC50 = 27 nM T65864 CUT1S8 71452133 IC50 = 12 nM T65864 C53GWF 71452135 IC50 = 220 nM T65864 CEBO91 71452977 IC50 > 10000 nM T65864 C52KFW 71453605 IC50 = 210 nM T65864 C9LWS3 71453606 IC50 = 15 nM T65864 CU4O2Q 71453607 IC50 = 35 nM T65864 C3AF9W 71453608 IC50 = 14 nM T65864 C9FQC8 71453609 IC50 = 120 nM T65864 CR1F0H 71453610 IC50 = 25 nM T65864 CE1PX3 71453733 IC50 = 11 nM T65864 CU07SO 71453962 IC50 = 3100 nM T65864 COU97C 71453963 IC50 = 4400 nM T65864 C4MIP0 71453964 IC50 = 220 nM T65864 C82FZD 71453965 IC50 = 11 nM T65864 C94IFE 71453966 IC50 = 10 nM T65864 C8QEP0 71453967 IC50 = 13 nM T65864 C31XLP 71453968 IC50 = 970 nM T65864 C9G2RF 71453969 IC50 = 850 nM T65864 C5DT4M 71454830 IC50 = 30 nM T65864 CPQE96 71454831 IC50 = 80 nM T65864 C1KYI8 71455335 IC50 = 130 nM T65864 CQK67Z 71455336 IC50 = 10 nM T65864 CW50OU 71455469 IC50 = 15 nM T65864 CWT08P 71455470 IC50 = 345 nM T65864 C0XJB7 71455705 IC50 = 9 nM T65864 C8NJ1X 71455706 IC50 = 12 nM T65864 C9C4GU 71455707 IC50 = 27 nM T65864 C23XFT 71455708 IC50 = 40 nM T65864 C8YJM0 71455709 IC50 = 6200 nM T65864 CMPD43 71455710 IC50 = 4700 nM T65864 C7FHJ9 71457109 IC50 = 40 nM T65864 C83MNK 71457110 IC50 = 180 nM T65864 C63EFT 71457111 IC50 = 200 nM T65864 C9TZK4 71457259 IC50 = 16 nM T65864 CI9B4S 71457484 IC50 = 30 nM T65864 CVP4H1 71457485 IC50 = 4 nM T65864 CUHA01 71457486 IC50 = 990 nM T65864 CB6K0P 71457487 IC50 = 17 nM T65864 C4J3IN 71457488 IC50 = 3800 nM T65864 CA8KT1 71457489 IC50 = 42 nM T65864 C76NGD 71458463 IC50 = 6700 nM T65864 C0D4PQ 71458977 IC50 = 36 nM T65864 C9UIP7 71458978 IC50 = 12 nM T65864 CL05AD 71458979 IC50 = 2000 nM T65864 CML63H 71458980 IC50 = 1500 nM T65864 CQN20S 71459107 IC50 = 2989 nM T65864 CVI6H7 71459354 IC50 = 29 nM T65864 CVT69Q 71459356 IC50 = 40 nM T65864 CHQZ25 71459584 IC50 > 10000 nM T65864 CSA71O 71460774 IC50 = 14 nM T65864 C5X8PM 71460775 IC50 = 24 nM T65864 CGD4C8 71460914 IC50 = 740 nM T65864 C4STL5 71460915 IC50 = 2600 nM T65864 C7VXY4 71461126 IC50 = 10 nM T65864 C9T5QS 71461127 IC50 = 3300 nM T65864 C4C5AG 71461128 IC50 = 3 nM T65864 C6KHP9 71461129 IC50 = 4800 nM T65864 C34FNC 71461131 IC50 = 84 nM T65864 C1FZH3 71462502 IC50 = 55 nM T65864 CZU37G 71462503 IC50 = 1200 nM T65864 CPXN98 71462610 IC50 = 290 nM T65864 CVI7X0 71462864 IC50 = 6800 nM T65864 CK3XZ9 71462865 IC50 = 83 nM T65864 CTA4K2 71462867 IC50 = 1600 nM T65864 CU47BO 71541785 IC50 = 4070 nM T65864 C4QC5N 71541791 IC50 = 5210 nM T65864 C7IWY9 71541886 IC50 = 16190 nM T65864 CPX50S 71543197 IC50 = 54310 nM T65864 CJ5O3G 71543200 IC50 = 14170 nM T65864 C9Z8AP 71543313 IC50 = 1603 nM T65864 CCZ7O8 71545200 IC50 = 11 nM T65864 C5ET0B 71545203 IC50 = 21 nM T65864 C8MNV5 71545204 IC50 = 2 nM T65864 CS7W6Q 71545205 IC50 = 27 nM T65864 CD37VJ 71545361 IC50 = 1 nM T65864 CHV87B 71545362 IC50 = 1 nM T65864 CV5J6Y 71545363 IC50 = 20 nM T65864 CYJ78S 71545364 IC50 = 2 nM T65864 C3W9ZG 71545365 IC50 = 1 nM T65864 CLO79S 71545520 IC50 = 0.3 nM T65864 CVFK78 71545521 IC50 = 0.7 nM T65864 C07XIK 71545522 IC50 = 2 nM T65864 CD63IG 71545523 IC50 = 7 nM T65864 C2KPN5 71545524 IC50 = 1 nM T65864 C98GPX 71545680 IC50 = 98 nM T65864 C6E1TI 71545681 IC50 = 12 nM T65864 CIC24O 71545682 IC50 = 220 nM T65864 C3ZC7X 71545683 IC50 = 4 nM T65864 C69GKW 71545684 IC50 = 0.5 nM T65864 C7XQE4 71545857 IC50 = 44 nM T65864 C8M7NB 71545858 IC50 = 3 nM T65864 CUL31Y 71545859 IC50 = 0.2 nM T65864 C3LK9W 71545860 IC50 = 10 nM T65864 C2VR9J 71545861 IC50 = 3 nM T65864 CAY4T0 71546016 IC50 = 89 nM T65864 C9P0NU 71546017 IC50 = 83 nM T65864 C86IHO 71546018 IC50 = 3 nM T65864 CT13PY 71546019 IC50 = 2 nM T65864 CT0OC8 71546020 IC50 = 54 nM T65864 CS4WB6 71546021 IC50 = 3 nM T65864 CKV1Z9 71546183 IC50 = 5 nM T65864 CJV69F 71546184 IC50 = 2 nM T65864 CLZ9D7 71546185 IC50 = 9 nM T65864 C6Z5KS 71546186 IC50 = 3 nM T65864 CNZL54 71546187 IC50 = 27 nM T65864 CHJ3Z2 71546356 IC50 = 19 nM T65864 CYD45I 71546357 IC50 = 6 nM T65864 C32DUX 71546358 IC50 = 5 nM T65864 C7LB0I 71546359 IC50 = 14 nM T65864 CWS3L1 71546360 IC50 = 7 nM T65864 CM9ZT4 71546524 IC50 = 94 nM T65864 CERQ05 71546525 IC50 = 160 nM T65864 CF1D2K 71546526 IC50 = 3 nM T65864 CEU93V 71546527 IC50 = 8 nM T65864 CMR1X7 71546528 IC50 = 29 nM T65864 CYZ7J2 71546529 IC50 = 210 nM T65864 C26BTI 71546681 IC50 = 1 nM T65864 CCN01X 71547862 IC50 > 10000 nM T65864 CB3SO2 71567006 IC50 > 10000 nM T65864 CDJY72 71568837 IC50 > 10000 nM T65864 CZ31PU 71583657 IC50 = 1700 nM T65864 CRC5M0 71605046 IC50 = 35 nM T65864 C7GN8S 71605048 IC50 = 35 nM T65864 CT90RH 71605222 IC50 = 24 nM T65864 CV47WL 71625692 IC50 = 4.3 nM T65864 C8SJX7 71625693 IC50 = 4.7 nM T65864 CL2A0I 71625803 IC50 = 20 nM T65864 C6GDA4 71625804 IC50 = 454 nM T65864 CTLG41 71625805 IC50 = 73 nM T65864 C6ZW1R 71714236 IC50 = 4 nM T65864 CKV91X 71714379 IC50 = 0.8 nM T65864 CHC8Q5 71714380 IC50 = 2.8 nM T65864 CAI68B 71714533 IC50 = 7.7 nM T65864 CXSI14 71718330 IC50 > 100000 nM T65864 C1TM3P 71720141 IC50 > 100000 nM T65864 CZAH39 71748684 IC50 = 1 nM T65864 C14BLE 72713331 IC50 = 63 nM T65864 CE7OH2 72713543 IC50 = 94 nM T65864 CY7FA2 72713544 IC50 = 87 nM T65864 C2Y8AB 72713545 IC50 = 34 nM T65864 CI5B2F 72713546 IC50 = 72 nM T65864 C2F5ML 72713547 IC50 = 571 nM T65864 C35OKU 72713548 IC50 = 563 nM T65864 C52ABZ 72713550 IC50 = 115 nM T65864 C5ES2C 72713551 IC50 = 122 nM T65864 C07NEJ 72713552 IC50 = 21 nM T65864 CD63JL 72713553 IC50 = 107 nM T65864 C6RK2D 72713765 IC50 = 481 nM T65864 CDO06G 72713766 IC50 = 25 nM T65864 CG3Z1F 72713767 IC50 = 42 nM T65864 C82CLY 72713769 IC50 = 218 nM T65864 CLO31X 72713770 IC50 = 132 nM T65864 C2RL4W 72713771 IC50 = 146 nM T65864 C82SHQ 72713772 IC50 = 207 nM T65864 CA6ED1 72713773 IC50 = 48 nM T65864 CY10WS 72713774 IC50 = 61 nM T65864 C3AFG5 72713775 IC50 = 233 nM T65864 COT2Y5 72713776 IC50 = 1060 nM T65864 C8AUB6 72713777 IC50 = 151 nM T65864 CUZX04 72713778 IC50 = 205 nM T65864 C51CQV 72713779 IC50 = 2430 nM T65864 CNWL94 72713780 IC50 = 4540 nM T65864 CW5D2Y 72713781 IC50 = 103 nM T65864 C2FX0D 72713782 IC50 = 7810 nM T65864 CJTH10 72713783 IC50 = 763 nM T65864 C8KIT1 72713978 IC50 = 33 nM T65864 CX9FN7 72713979 IC50 = 147 nM T65864 C5QCO7 72713980 IC50 = 41 nM T65864 CW7Q6M 72713981 IC50 = 85 nM T65864 C5ZYV0 72713982 IC50 = 160 nM T65864 C1VPY8 72713983 IC50 = 557 nM T65864 C6G2OU 72713984 IC50 = 79 nM T65864 C2ZE7R 72713985 IC50 = 18570 nM T65864 CY5G2X 72713986 IC50 = 20 nM T65864 C4E5UD 72713987 IC50 = 631 nM T65864 CTQ7I0 72713988 IC50 = 22 nM T65864 CJL83X 72713989 IC50 = 280 nM T65864 C3TK8O 72713990 IC50 = 28 nM T65864 CUD5N1 72713991 IC50 = 819 nM T65864 C56YBV 72713997 IC50 = 3 nM T65864 CG91JM 72713998 IC50 = 1.7 nM T65864 C4Z8HO 72714202 IC50 = 53 nM T65864 C4FN8L 72714204 IC50 = 516 nM T65864 CHM8T6 72714205 IC50 = 28190 nM T65864 CLBZ26 72714206 IC50 = 21 nM T65864 C5KJ8H 72714211 IC50 > 10000 nM T65864 C0NQ5X 72714212 IC50 > 10000 nM T65864 C5QBV7 72714213 IC50 = 1944 nM T65864 C0B4PF 72714222 IC50 = 17 nM T65864 CP9LH4 72714223 IC50 = 10 nM T65864 C6G2XJ 72714224 IC50 = 25 nM T65864 C8OY6Q 76310785 IC50 = 2480 nM T65864 C60COV 76310786 IC50 = 590 nM T65864 CAQ90E 76310787 IC50 = 1400 nM T65864 CAL3U7 76310788 IC50 = 140 nM T65864 CBG94X 76310789 IC50 = 2170 nM T65864 C12YAE 76314414 IC50 = 783 nM T65864 C9K4WT 76314416 IC50 = 430 nM T65864 CNP2Z9 76314417 IC50 = 730 nM T65864 CZ2GV7 76314418 IC50 = 290 nM T65864 COH59Y 76314419 IC50 = 3800 nM T65864 C1LZA4 76317974 IC50 = 23500 nM T65864 CJ2Y6E 76317975 IC50 = 11400 nM T65864 C3AGC7 76317976 IC50 = 460 nM T65864 C70IFZ 76317977 IC50 = 1170 nM T65864 C97RBS 76317979 IC50 = 96 nM T65864 C0V4QA 76317980 IC50 = 4200 nM T65864 CC65HR 76317982 IC50 = 190 nM T65864 C25TDN 76321242 IC50 = 196 nM T65864 COD90K 76321706 IC50 = 19500 nM T65864 CVG6O5 76321707 IC50 = 6510 nM T65864 C1BW8J 76321709 IC50 = 11200 nM T65864 C1G9AH 76321710 IC50 = 11600 nM T65864 C1AI0J 76325315 IC50 = 140 nM T65864 CM8I4T 76325316 IC50 = 380 nM T65864 C3U9VE 76325317 IC50 = 1790 nM T65864 CMWJ79 76325318 IC50 = 400 nM T65864 COC52I 76325319 IC50 = 5730 nM T65864 C6MDE5 76325320 IC50 = 740 nM T65864 CL49QH 76325321 IC50 = 3200 nM T65864 CPQA45 76325323 IC50 = 345 nM T65864 C20SAY 76325325 IC50 = 56000 nM T65864 CXEL67 76325326 IC50 = 990 nM T65864 C25UVD 76325327 IC50 > 100000 nM T65864 C5LB1T 76325328 IC50 = 710 nM T65864 CM35GK 76325329 IC50 = 1190 nM T65864 CI85VP 76325330 IC50 = 12500 nM T65864 COI2P8 76328018 IC50 = 1.8 nM T65864 CT2U7G 76328019 IC50 = 1.6 nM T65864 CU0NK1 76328020 IC50 = 665 nM T65864 C7M3YJ 76328868 IC50 > 100000 nM T65864 C1OT8R 76332536 IC50 = 158000 nM T65864 CO07HT 76332537 IC50 = 1440 nM T65864 CRA79N 76332538 IC50 = 1490 nM T65864 CJG48Z 76332539 IC50 = 430 nM T65864 CB5Y0Z 76332540 IC50 = 185 nM T65864 CSG89Y 76332541 IC50 = 250 nM T65864 CDY62X 76332543 IC50 = 890 nM T65864 C6DZ3T 76332544 IC50 = 2400 nM T65864 C5CE6Y 76332545 IC50 = 1590 nM T65864 CI91LV 76332547 IC50 = 5180 nM T65864 C3G1XK 76335725 IC50 = 65 nM T65864 CHX67J 76336155 IC50 = 1870 nM T65864 CDC82P 76336156 IC50 = 2300 nM T65864 CE97SW 76336158 IC50 = 91 nM T65864 CJ50KE 76336159 IC50 = 1530 nM T65864 CUYT59 78319219 IC50 = 5110 nM T65864 CPG3A5 86302574 IC50 > 30000 nM T65864 C1HW4B 89735655 IC50 > 100000 nM T65864 CY0UC4 90645194 IC50 > 10000 nM T65864 C67BLK 90656196 IC50 > 10000 nM T65864 C39FOS 90656197 IC50 > 10000 nM T65864 C2QW6F 90656198 IC50 > 10000 nM T65864 CDUS92 90656199 IC50 > 10000 nM T65864 CIP5Q8 90656200 IC50 > 10000 nM T65864 C3O5BS 90656201 IC50 > 10000 nM T65864 C6FB0V 90656202 IC50 = 5210 nM T65864 C2K0XC 90656203 IC50 = 3770 nM T65864 C0CEV3 90656204 IC50 = 2830 nM T65864 C31QUS 90656205 IC50 = 1490 nM T65864 C4TAB6 90656206 IC50 = 1050 nM T65864 CA9H7B 90656207 IC50 > 10000 nM T65864 CW65FA 90656208 IC50 > 10000 nM T65864 CMH6T8 90664306 IC50 > 1600 nM T65864 C8GX5H 90665650 IC50 = 460 nM T65864 CP9I5F 90665651 IC50 = 310 nM T65864 C24PHD 90665652 IC50 = 38 nM T65864 CFH74I 90665653 IC50 = 1500 nM T65864 CKPG46 90666065 IC50 = 83 nM T65864 CF95HX 90666066 IC50 = 46 nM T65864 C09XAJ 90666067 IC50 = 46 nM T65864 C5VIB9 90666068 IC50 = 140 nM T65864 C1O7KT 90666069 IC50 = 29 nM T65864 C1I5JK 90666070 IC50 = 20 nM T65864 CQ1RN2 90666071 IC50 = 115 nM T65864 CX6D4L 90666072 IC50 = 36 nM T65864 C5XYV9 90666073 IC50 = 337 nM T65864 CI1F9V 90666074 IC50 = 498 nM T65864 CA86DM 90666075 IC50 = 173 nM T65864 C2JCV6 90666076 IC50 = 411 nM T65864 C2JRE9 90666077 IC50 = 186 nM T65864 CR30QC 90666078 IC50 = 430 nM T65864 C7N6SR 90666079 IC50 = 396 nM T65864 CO75JN 90666241 IC50 = 20 nM T65864 CY1E3X 90666242 IC50 = 44 nM T65864 CL3S4Z 90666343 IC50 = 70 nM T65864 C0Y8ZK 91933875 IC50 > 1000 nM T65864 C6ZFW9 101913690 IC50 = 30 nM T65864 C9VSP7 101913691 IC50 = 34 nM T65864 C61FOL 118144367 IC50 = 3623 nM T65864 CG7QL4 118705925 IC50 = 571 nM T65864 CY7BI2 118706214 IC50 > 10000 nM T65864 CK1HA9 118706303 IC50 = 1310 nM T65864 C35UDW 118706304 IC50 = 1210 nM T65864 CZ1I4D 118706305 IC50 = 23 nM T65864 CAC09F 118706306 IC50 = 23.4 nM T65864 C4R8VS 118706307 IC50 = 271 nM T65864 C2C0AG 118707521 IC50 = 1020 nM T65864 C2DJA0 118707522 IC50 = 2510 nM T65864 CBF28W 118707523 IC50 = 250 nM T65864 CQ6ON4 118707525 IC50 = 12000 nM T65864 C38UWP 118707526 IC50 > 100000 nM T65864 C64ZQX 118707543 IC50 = 82100 nM T65864 C3R7XB 118725448 IC50 = 2400 nM T65864 CJT49C 118725449 IC50 = 2000 nM T65864 CG4W6V 118725450 IC50 = 1700 nM T65864 CT4WP3 118725451 IC50 = 450 nM T65864 C3SAQ6 118725452 IC50 = 560 nM T65864 CQ6HI7 118725453 IC50 = 2800 nM T65864 C4X9CT 118725454 IC50 = 2500 nM T65864 CA17EJ 118725455 IC50 = 15 nM T65864 CH1I7T 118725456 IC50 < 46 nM T65864 CC80JT 118725457 IC50 > 10000 nM T65864 CV05IX 118725458 IC50 = 490 nM T65864 C5TO3U 118725459 IC50 = 190 nM T65864 CD34GN 118725460 IC50 = 86 nM T65864 CAS6N4 118725461 IC50 = 390 nM T65864 CA1PU9 118725462 IC50 = 270 nM T65864 CPVI19 118725463 IC50 = 53 nM T65864 C2NQ1T 118725464 IC50 = 76 nM T65864 CZ82KA 118725885 IC50 = 642 nM T65864 CSV5K7 118725886 IC50 = 297 nM T65864 C9XV2B 118725887 IC50 = 140 nM T65864 C6KCQ9 118725888 IC50 = 1666 nM T65864 C6LCD8 118725889 IC50 = 36 nM T65864 CI96GZ 118725890 IC50 = 246 nM T65864 CL3KT6 118725891 IC50 = 1699 nM T65864 C2JNF8 118725892 IC50 = 191 nM T65864 CU9KV7 118725893 IC50 = 335 nM T65864 C51HGX 118725894 IC50 = 123 nM T65864 C3HP6G 118725895 IC50 = 211 nM T65864 CR4K1M 118725896 IC50 = 164 nM T65864 C95CUL 118725897 IC50 = 165 nM T65864 CN27BI 118725898 IC50 = 39 nM T65864 CH1VK2 118725899 IC50 = 223 nM T65864 C5IM2Q 118725900 IC50 = 723 nM T65864 CP7DK8 118725901 IC50 = 416 nM T65864 CL8W3Q 118725902 IC50 = 764 nM T65864 CNL1Z4 118725903 IC50 = 135 nM T65864 C5S2OE 118725904 IC50 = 612 nM T65864 CL0CJ2 118725905 IC50 = 451 nM T65864 C4UTF5 118725906 IC50 = 2184 nM T65864 C4PQ8K 118725907 IC50 = 655 nM T65864 CE7ZH9 118725908 IC50 = 208 nM T65864 CM7IQ3 118725909 IC50 = 356 nM T65864 C3WF5U 118725910 IC50 = 153 nM T65864 CGR19E 118725911 IC50 = 128 nM T65864 CZ8RX6 118725912 IC50 = 146 nM T65864 CU9RB6 118725913 IC50 = 354 nM T65864 CBO8S2 118725914 IC50 = 181 nM T65864 C5CMS9 118725915 IC50 = 36 nM T65864 CEJ7T0 118725916 IC50 = 146 nM T65864 CHB9S7 118959070 IC50 > 120000 nM T65864 CV5F2D 118959076 IC50 = 100000 nM T65864 C8L1QI 118959080 IC50 > 120000 nM T65864 CX9N1Q 118959089 IC50 > 120000 nM T65864 CO2L3G 118959104 IC50 = 35000 nM T65864 C5GLM2 121232441 IC50 = 7 nM T65864 C9CV7H 121411850 IC50 < 100 nM T65864 CU3BI0 121412063 IC50 < 100 nM T65864 C2TSV7 122177851 IC50 = 35 nM T65864 CEK9S7 122177852 IC50 = 66 nM T65864 C40APN 122177853 IC50 = 87 nM T65864 CCN6F5 122177854 IC50 = 4.5 nM T65864 CE68SL 122177855 IC50 = 54 nM T65864 CSFJ19 122177913 IC50 = 6.5 nM T65864 C53NSH 122177914 IC50 = 4.3 nM T65864 CJD03F 122177915 IC50 = 5.6 nM T65864 CX8JI0 122177916 IC50 = 3.7 nM T65864 CJI3N8 122177917 IC50 = 4.6 nM T65864 CJHF98 122177918 IC50 = 354 nM T65864 CU15EY 122177919 IC50 = 56 nM T65864 CGDL13 122177920 IC50 = 77 nM T65864 CVE19K 122177921 IC50 = 345 nM T65864 CB1HF0 122177922 IC50 = 34 nM T65864 CER2Y0 122177923 IC50 = 23 nM T65864 COQ7U6 122177924 IC50 = 345 nM T65864 CV1A2F 122177925 IC50 = 4.7 nM T65864 CJ6RM1 122177926 IC50 = 4.5 nM T65864 CC13JY 122177927 IC50 = 44 nM T65864 CZQO07 122196303 IC50 = 399 nM T65864 C7LR8Z 122196304 IC50 = 766 nM T65864 CGK94L 122196305 IC50 = 209 nM T65864 CE6UA3 122196306 IC50 = 251 nM T65864 CBXL72 122196307 IC50 = 171 nM T65864 C5J0HO 122196308 IC50 > 10000 nM T65864 C6YSR2 122196309 IC50 > 10000 nM T65864 COY82I 122196310 IC50 = 2040 nM T65864 C0KE4Y 122196311 IC50 = 3370 nM T65864 CMWG96 122196359 IC50 = 1240 nM T65864 CU6L5G 122196360 IC50 = 1480 nM T65864 CCA29B 122196361 IC50 = 1810 nM T65864 C6UY2L 122633880 IC50 = 89 nM T65864 CC7P2W 122633900 IC50 = 106 nM T65864 CN41IF 122634050 IC50 = 62 nM T65864 C3NHU5 127030449 IC50 = 8 nM T65864 CI73JH 127030772 IC50 = 33 nM T65864 CEI25F 127030791 IC50 = 6 nM T65864 CUQ5T4 127030792 IC50 = 18 nM T65864 C7Q6PH 127030793 IC50 = 24 nM T65864 CRO3B9 127031107 IC50 = 123 nM T65864 CXV6F2 127031108 IC50 = 6 nM T65864 C90LYU 127031109 IC50 = 13 nM T65864 CD5A9R 127031117 IC50 = 9 nM T65864 CV7KB9 127031414 IC50 = 25 nM T65864 CANH59 127031725 IC50 = 27 nM T65864 C3UDF1 127034594 IC50 = 167 nM T65864 CG68HZ 127039911 IC50 = 370 nM T65864 CR5D0T 127041573 IC50 = 2700 nM T65864 CA43DP 127052672 IC50 > 5000 nM T65864 C9TQG2 127052673 IC50 > 5000 nM T65864 CG3W6F 129900105 IC50 = 463.8 nM T65864 CVE3W1 129900106 IC50 = 0.6 nM T65864 C71KMN 130429150 IC50 = 9221 nM T65864 CSG8J3 130429224 IC50 > 50000 nM T65864 C5PT1M 130429242 IC50 = 27143 nM T65864 C0UNO3 130429244 IC50 > 100000 nM T65864 CGFK71 130429248 IC50 = 20517 nM T65864 CEX8D1 130429250 IC50 = 8815 nM T65864 C9J6ZK 130429255 IC50 > 50000 nM T65864 C51EID 132496692 IC50 = 2 nM T65864 CKFI10 134141966 IC50 = 44 nM T65864 CI9QD8 134143410 IC50 = 46 nM T65864 C8WZ1F 134151653 IC50 = 899 nM T65864 C5HA8K 134610596 IC50 = 93200 nM T65864 C2AN7T 134611886 IC50 > 100000 nM T65864 C54FXD 134957362 IC50 > 10000 nM T65864 C8GZ2B 135449326 Ki > 4000 nM T65864 C0SCD8 135470346 IC50 = 560 nM T65864 CM2UH4 135894362 IC50 > 1000 nM T65864 CY19DW 135894364 IC50 > 1000 nM T65864 C61KVL 135930668 EC50 = 5200 nM T65864 C72CDP 135930669 EC50 <= 7 nM T65864 CHA4N2 136013680 IC50 > 10 nM T65864 CVIC49 136069671 IC50 = 8700 nM T65864 CT6P2Z 136126660 Ki = 49 nM T65864 CKC54E 136126661 Ki = 4.7 nM T65864 CM4KA6 136126662 Ki = 6.8 nM T65864 C1T3VA 136126663 Ki = 2.9 nM T65864 C5AKQ2 136146217 IC50 = 60 nM T65864 CZ7EX0 136183413 IC50 > 30000 nM T65864 CFC86W 136193077 IC50 = 80 nM T65864 C15HQK 136218656 IC50 > 1000 nM T65864 CZ06UK 136218660 IC50 > 1000 nM T65864 CML48X 136218661 IC50 > 1000 nM T65864 COB69I 136218662 IC50 > 1000 nM T65864 CSL6Q8 136218663 IC50 > 1000 nM T65864 C1YUD0 136219394 IC50 > 10 nM T65864 CTFJ83 136226213 IC50 > 1000 nM T65864 C5QAT2 136236302 IC50 = 3 nM T65864 C5EV8A 136240902 IC50 > 1000 nM T65864 CX9LB5 136240903 IC50 > 1000 nM T65864 CMC58H 136240944 IC50 > 1000 nM T65864 C60PRZ 136241012 IC50 > 1000 nM T65864 C1UL0F 136242884 IC50 = 8.4 nM T65864 C1Q9YN 136252259 IC50 > 1000 nM T65864 CIU8W3 136254389 IC50 > 10 nM T65864 C5JIR2 136987005 IC50 = 95.5 nM T65864 COI75S 137348574 IC50 = 1 nM T65864 C86OQA 137348940 IC50 = 5.4 nM T65864 CAM8H7 137631669 IC50 = 4.7 nM T65864 C0QBR8 137631695 IC50 = 6.7 nM T65864 CJA4G6 137631710 IC50 = 2.6 nM T65864 CH9O7Z 137631713 IC50 = 38 nM T65864 CP8K3J 137632201 IC50 = 0.2 nM T65864 C9KY3F 137632254 IC50 = 60.2 nM T65864 CMG41Z 137632321 IC50 = 32.9 nM T65864 CS4V5P 137632440 IC50 = 5.2 nM T65864 C3JGA9 137632725 IC50 = 1.6 nM T65864 CSB1X0 137633255 IC50 = 13.1 nM T65864 C67ACU 137633444 IC50 = 129.3 nM T65864 CV2ZY8 137633566 IC50 = 59.3 nM T65864 C2PMQ0 137635421 IC50 = 0.1 nM T65864 C4W5HN 137635818 IC50 = 0.6 nM T65864 C23WJU 137635942 IC50 = 4.2 nM T65864 C1SI0V 137636154 IC50 = 5.4 nM T65864 C4V1EU 137636264 IC50 = 35 nM T65864 CXLM63 137636621 IC50 = 4 nM T65864 C8GQD5 137636872 IC50 > 10000 nM T65864 C64WAG 137637444 IC50 = 40.9 nM T65864 C1G6KJ 137637551 IC50 = 0.8 nM T65864 CG4TJ6 137638097 IC50 = 3 nM T65864 C4NBP2 137638482 IC50 = 1 nM T65864 COD2C5 137638574 IC50 = 0.4 nM T65864 CDHR26 137638664 IC50 = 288 nM T65864 CLGH04 137638967 IC50 = 100 nM T65864 CLM2E7 137639118 IC50 = 214 nM T65864 CHGX21 137639663 IC50 = 0.6 nM T65864 C6NPM1 137639803 IC50 = 23.8 nM T65864 CNE0Z1 137639840 IC50 = 4 nM T65864 CS3RQ4 137639936 IC50 = 26 nM T65864 CPB36N 137640949 IC50 = 1.6 nM T65864 CIAX13 137641023 IC50 = 0.28 nM T65864 CT38UG 137641182 IC50 = 17 nM T65864 CY71MB 137641325 IC50 = 0.2 nM T65864 C3M0AT 137642113 IC50 = 0.4 nM T65864 CG0P7F 137642583 IC50 = 2 nM T65864 C0F3OK 137642727 IC50 = 32.5 nM T65864 C53RLU 137642863 IC50 = 1.3 nM T65864 C6QL2D 137642948 IC50 = 0.4 nM T65864 CYL1R5 137643579 IC50 = 2 nM T65864 CSYL15 137644166 IC50 = 969 nM T65864 CNK3C1 137644195 IC50 = 12 nM T65864 C2L8WJ 137644650 IC50 = 2.4 nM T65864 CGR1Y5 137644830 IC50 = 5 nM T65864 C2J5LE 137645653 IC50 = 2300.8 nM T65864 CW3IE6 137645681 IC50 = 17 nM T65864 CAY2W4 137646016 IC50 = 1952 nM T65864 CFO76I 137646540 IC50 = 182.3 nM T65864 CGNM85 137646697 IC50 = 3 nM T65864 C8O0BX 137647038 IC50 = 5.3 nM T65864 CPWT95 137647219 IC50 = 2 nM T65864 C6YXV2 137647333 IC50 = 1.2 nM T65864 C6HAS1 137647418 IC50 = 2.7 nM T65864 CMON76 137647931 IC50 = 0.4 nM T65864 CI2K4X 137648079 IC50 = 374.4 nM T65864 CFX52L 137649093 IC50 = 2.6 nM T65864 C70VNG 137649240 IC50 = 1.1 nM T65864 C5UE8A 137649558 IC50 = 241 nM T65864 C8DAQ1 137649779 IC50 = 0.5 nM T65864 CGNK76 137650697 IC50 = 0.6 nM T65864 CN13EH 137650943 IC50 = 36 nM T65864 CTQJ93 137650950 IC50 = 382.4 nM T65864 CNC20A 137650995 IC50 = 35.7 nM T65864 CCO1Q7 137651285 IC50 = 13.1 nM T65864 CL6A5T 137651622 IC50 = 0.8 nM T65864 CD1Z9I 137651824 IC50 = 106.7 nM T65864 C1TMW8 137651977 IC50 = 1 nM T65864 C3DF4I 137652013 IC50 = 1.4 nM T65864 C3P4LM 137652106 IC50 = 1.3 nM T65864 CLN2U7 137652270 IC50 = 710 nM T65864 CCTP83 137652548 IC50 = 17.6 nM T65864 CLN2M3 137652755 IC50 = 126 nM T65864 C59KAW 137653285 IC50 = 0.8 nM T65864 CV8P0Z 137653773 IC50 = 0.9 nM T65864 CKJ17T 137654104 IC50 = 0.4 nM T65864 C8MH2Z 137654276 IC50 = 217 nM T65864 CW0S8M 137654802 IC50 = 10.9 nM T65864 CMJF60 137655822 IC50 = 3 nM T65864 CPY1U3 137656311 IC50 = 22 nM T65864 C2QS9U 137656461 IC50 = 1.2 nM T65864 CMJ6C1 137656574 IC50 = 34.9 nM T65864 CY2QT7 137656905 IC50 = 0.6 nM T65864 CBHO36 137657256 IC50 = 659.1 nM T65864 C51LSJ 137657279 IC50 = 4.8 nM T65864 CBI64H 137657498 IC50 = 149 nM T65864 COW4X5 137657506 IC50 = 0.2 nM T65864 CV1WJ5 137657591 IC50 = 137.8 nM T65864 C10NJC 137657604 IC50 = 19.3 nM T65864 CW91OB 137657852 IC50 = 1.3 nM T65864 CDMX65 137658488 IC50 = 0.7 nM T65864 CH5JU3 137658981 IC50 = 7 nM T65864 CZFJ89 137660093 IC50 > 10000 nM T65864 C10PNV 137660797 IC50 = 0.3 nM T65864 CA3XC2 137660956 IC50 = 5920 nM T65864 CW0Q7M 137661455 IC50 = 0.3 nM T65864 CS32IR 137661932 IC50 = 47 nM T65864 CH2T5R 139030330 IC50 = 26 nM T65864 C7JEX9 139030331 IC50 = 18 nM T65864 COE1X5 139030332 IC50 = 71 nM T65864 CM3A8O 139030333 IC50 = 3.7 nM T65864 CX5AV4 145505929 IC50 = 12 nM T65864 COUM49 145506081 IC50 = 14 nM T65864 CT6WU5 145506114 IC50 = 210 nM T65864 C1KQ6Y 145506115 IC50 = 11 nM T65864 C6VB3O 145925651 IC50 >= 5000 nM T65864 CI1VH9 145985185 IC50 > 200000 nM T65864 CGZ76S 145986724 IC50 = 26 nM T65864 CNLH48 145988888 IC50 > 200000 nM T65864 CRT48W 145993502 IC50 > 200000 nM T65864 C42BWS 145994862 IC50 = 55 nM T65864 CUH9P6 155077159 IC50 = 16 nM T65864 CY1ZH2 155510358 IC50 = 22 nM T65864 CV0MZ9 155510817 IC50 = 15 nM T65864 CXWI87 155511357 IC50 = 81 nM T65864 CO5WR4 155511447 IC50 = 18 nM T65864 CH9N0J 155511915 IC50 > 500 nM T65864 CY1VF8 155511959 IC50 = 370 nM T65864 CD8M7Q 155512392 IC50 = 20 nM T65864 CHEI63 155513115 IC50 > 500 nM T65864 C2MD1Q 155513187 IC50 > 10000 nM T65864 C09TIS 155513203 IC50 = 280 nM T65864 C4PDT6 155514077 IC50 = 45 nM T65864 CD0SG7 155514146 IC50 > 10000 nM T65864 CT5YG4 155514435 IC50 = 44 nM T65864 CWBU69 155514452 IC50 = 91 nM T65864 C6ZUK4 155514537 IC50 = 260 nM T65864 C6SQX5 155514684 IC50 = 28 nM T65864 C9O1QE 155515323 IC50 > 500 nM T65864 CP4UQ3 155515929 IC50 = 15 nM T65864 CM3E4T 155516307 IC50 = 4005 nM T65864 CA54SV 155516886 IC50 = 14 nM T65864 CL7G5U 155517186 IC50 > 10000 nM T65864 CFG2M8 155517577 IC50 = 9 nM T65864 CT24JB 155517821 IC50 > 30000 nM T65864 C12DHX 155517839 IC50 > 10000 nM T65864 C0HZ8O 155518052 IC50 > 500 nM T65864 CR1A0B 155518258 IC50 > 10000 nM T65864 C86HPW 155518524 IC50 = 88000 nM T65864 CFD86N 155518907 IC50 = 4400 nM T65864 CNE3Q5 155519237 IC50 > 500 nM T65864 C68LNI 155519614 IC50 = 280 nM T65864 C2YQ5I 155519636 IC50 > 500 nM T65864 CD7JR5 155520366 IC50 = 14400 nM T65864 CU64PX 155520421 IC50 = 580 nM T65864 CUK59T 155520576 IC50 = 17 nM T65864 C0NMJ7 155520623 IC50 = 29 nM T65864 CLH7Y2 155520781 IC50 > 500 nM T65864 C86ALD 155521765 IC50 = 3 nM T65864 CIK2W8 155522314 IC50 = 16 nM T65864 CJ6Y8X 155522691 IC50 = 12300 nM T65864 CHF31J 155522721 IC50 = 1851 nM T65864 C6Z2QE 155522907 IC50 = 47 nM T65864 CQW9M3 155523312 IC50 = 61 nM T65864 C9NM7B 155523411 IC50 = 19 nM T65864 C92VJW 155523476 IC50 = 1170 nM T65864 CM2QO4 155523988 IC50 > 500 nM T65864 CV8P9Q 155524146 IC50 = 184 nM T65864 CYI5Z3 155524399 IC50 = 120 nM T65864 CP4L8F 155524599 IC50 > 10000 nM T65864 CH95PJ 155524845 IC50 > 500 nM T65864 CRG17A 155524993 IC50 = 2330 nM T65864 CW3S9D 155525178 IC50 = 19 nM T65864 CW96RL 155525249 IC50 > 10000 nM T65864 C5E4WZ 155525348 IC50 > 500 nM T65864 C8N9QV 155525434 IC50 > 30000 nM T65864 CEIW40 155525530 IC50 = 7 nM T65864 CF4MP8 155525636 IC50 = 8540 nM T65864 C0S7GV 155525697 IC50 > 10000 nM T65864 C4F9QH 155525702 IC50 = 2350 nM T65864 C9HKF7 155526015 IC50 = 19 nM T65864 C3V8RW 155526111 IC50 = 59 nM T65864 C2Z1AW 155526520 IC50 = 360 nM T65864 CCGD64 155526869 IC50 = 20 nM T65864 C98ACB 155526885 IC50 = 2400 nM T65864 CLT3E4 155527966 IC50 = 987 nM T65864 CPW6E9 155528043 IC50 > 10000 nM T65864 CPEU39 155528262 IC50 = 3800 nM T65864 CYQ1E0 155528481 IC50 > 500 nM T65864 CEXY67 155528636 IC50 = 16 nM T65864 CQT70J 155529207 IC50 > 500 nM T65864 CXFH38 155529296 IC50 = 15 nM T65864 CO2JD6 155529363 IC50 > 500 nM T65864 C6ATZ2 155530054 IC50 > 500 nM T65864 CU9B7D 155530528 IC50 = 763 nM T65864 C58LZX 155531251 IC50 = 88 nM T65864 C0SR3H 155531653 IC50 > 500 nM T65864 CY6BV8 155531715 IC50 = 1290 nM T65864 C0QO5E 155531724 IC50 = 38 nM T65864 C54ARD 155532371 IC50 = 34500 nM T65864 C48FKU 155533602 IC50 > 500 nM T65864 C10DMX 155534844 IC50 > 10000 nM T65864 CLZ32Q 155534860 IC50 = 258 nM T65864 C6UDV1 155536548 IC50 = 20 nM T65864 CMW7K0 155536680 IC50 = 480 nM T65864 CQ39BV 155536797 IC50 = 13 nM T65864 CZ5A1P 155536847 IC50 > 500 nM T65864 CE7X0S 155536957 IC50 > 10000 nM T65864 C2CG1A 155537016 IC50 > 10000 nM T65864 CFC3D2 155537268 IC50 = 19 nM T65864 C9TXU8 155537377 IC50 = 158 nM T65864 C24SFW 155537433 IC50 > 500 nM T65864 C3ZHC0 155537470 IC50 = 24 nM T65864 C7WP5T 155537497 IC50 = 2440 nM T65864 C2A9KV 155537532 IC50 = 42 nM T65864 CD4G8Y 155538105 IC50 > 10000 nM T65864 CWP49G 155538536 IC50 > 500 nM T65864 COE67I 155538620 IC50 = 18 nM T65864 CEP37L 155538694 IC50 = 18 nM T65864 C6RD2N 155538801 IC50 > 500 nM T65864 CS4W6B 155538942 IC50 = 13 nM T65864 C46ICV 155539003 IC50 = 320 nM T65864 CBQ1O4 155539034 IC50 = 9460 nM T65864 C9UZJ6 155539371 IC50 = 24 nM T65864 C4LAT3 155539976 IC50 > 10000 nM T65864 CRKI54 155540083 IC50 = 6060 nM T65864 CW5U2N 155540164 IC50 > 30000 nM T65864 C5ORP4 155540981 IC50 > 10000 nM T65864 CIRG96 155541302 IC50 = 515 nM T65864 CBM39S 155541324 IC50 = 30 nM T65864 C32CFS 155541434 IC50 = 89 nM T65864 CAJ90M 155541538 IC50 = 12215 nM T65864 C8K3WL 155541562 IC50 = 27 nM T65864 C0M5HY 155541829 IC50 > 10000 nM T65864 C9ML7T 155541864 IC50 = 148 nM T65864 CMK7O9 155541940 IC50 > 10000 nM T65864 C3J8SM 155542090 IC50 = 88 nM T65864 C2S3FB 155542512 IC50 > 500 nM T65864 CA5UN7 155542968 IC50 = 280 nM T65864 C4KMP8 155543427 IC50 = 27 nM T65864 CGR9U1 155543795 IC50 > 30000 nM T65864 CQMZ76 155544092 IC50 > 10000 nM T65864 CWE36U 155544099 IC50 = 360 nM T65864 CI63KH 155544112 IC50 > 30000 nM T65864 CMS7U8 155544549 IC50 = 7040 nM T65864 C15KRU 155545689 IC50 = 2040 nM T65864 CUF13E 155546010 IC50 > 10000 nM T65864 CQ97ZD 155546227 IC50 > 500 nM T65864 CC9LQ2 155546287 IC50 = 13000 nM T65864 C36BPF 155546292 IC50 = 31 nM T65864 CT2S7A 155546431 IC50 > 10000 nM T65864 CX9WQ7 155546694 IC50 = 899 nM T65864 C1FKM7 155546916 IC50 > 500 nM T65864 CRVN92 155547073 IC50 = 4840 nM T65864 CMT19E 155547765 IC50 = 10 nM T65864 CY96SD 155548355 IC50 > 500 nM T65864 CW4LO3 155548563 IC50 = 250 nM T65864 CT07RL 155548603 IC50 = 470 nM T65864 C0X5EB 155549123 IC50 = 316 nM T65864 CIQM72 155549185 IC50 > 500 nM T65864 CB76ET 155549375 IC50 = 101 nM T65864 CK9Z5W 155550010 IC50 > 500 nM T65864 C8PA6D 155550766 IC50 = 23 nM T65864 C26ILZ 155551090 IC50 = 53 nM T65864 CR0K3W 155551204 IC50 > 500 nM T65864 C2REF6 155551339 IC50 = 2830 nM T65864 CZ9Y5A 155551667 IC50 > 10000 nM T65864 C75MHC 155551790 IC50 = 1520 nM T65864 C2FI6S 155552437 IC50 = 2220 nM T65864 C18YHM 155552761 IC50 = 6065 nM T65864 CAQU49 155552777 IC50 > 500 nM T65864 C7I9ER 155553064 IC50 > 500 nM T65864 C9C4XO 155553435 IC50 = 41 nM T65864 CE01LF 155553747 IC50 = 8120 nM T65864 CEBV41 155554010 IC50 = 55 nM T65864 C3I6NL 155554624 IC50 = 41 nM T65864 C0ZO6N 155555559 IC50 > 30000 nM T65864 C3JG0R 155555727 IC50 = 7700 nM T65864 CV60MW 155555951 IC50 = 22 nM T65864 CDC59Q 155556256 IC50 = 17 nM T65864 C9M4DG 155557125 IC50 = 29 nM T65864 C1AIF0 155557307 IC50 > 500 nM T65864 CAXC54 155558046 EC50 = 1940 nM T65864 CF1TN3 155558413 IC50 > 30000 nM T65864 CND16A 155558659 IC50 > 500 nM T65864 C5JRG0 155558848 IC50 = 50 nM T65864 CP18NC 155559676 IC50 = 117 nM T65864 CPOV46 155560224 IC50 > 500 nM T65864 CNX32F 155560561 IC50 = 27 nM T65864 CT39UJ 155561412 IC50 = 210 nM T65864 C10FWR 155561550 IC50 > 500 nM T65864 C6D7OT 155562118 IC50 > 10000 nM T65864 CUL57N 155562188 IC50 > 500 nM T65864 CQ6P4J 155562494 IC50 > 10000 nM T65864 C2EZX3 155562891 IC50 = 14350 nM T65864 CRC25F 155563369 IC50 = 21 nM T65864 CV1SK7 155563610 IC50 > 500 nM T65864 C0WCO2 155563644 IC50 = 513 nM T65864 CPS4C6 155563814 IC50 > 10000 nM T65864 C31SXI 155563958 IC50 = 40 nM T65864 C16JFY 155563983 IC50 > 10000 nM T65864 C8N2FR 155564003 IC50 = 400 nM T65864 C1DM5X 155564336 IC50 = 48 nM T65864 C8MOL1 155564646 IC50 = 6500 nM T65864 C0P7QO 155565131 IC50 > 500 nM T65864 C5YXO3 155565855 IC50 > 500 nM T65864 C4XT0Y 155565999 IC50 > 500 nM T65864 CLA4I9 155566444 IC50 > 500 nM T65864 CWGZ76 155566793 IC50 = 504 nM T65864 C6QY8E 155567320 IC50 = 831 nM T65864 CHZB01 155567574 IC50 > 500 nM T65864 CGX17T 155567824 IC50 = 44 nM T65864 CLG3Y8 155568520 IC50 > 500 nM T65864 CRD24F 155568639 IC50 = 51 nM T65864 C5P6AF 155568803 IC50 > 500 nM T65864 CZBS25 155568984 IC50 = 36 nM T65864 CWE74H 155569551 IC50 = 5800 nM T65864 C2Q6AH 155569559 IC50 = 7 nM T65864 C3CYJ6 135755216 IC50 = 8 nM T65864 C7UTN0 135899462 IC50 = 59 nM T65864 D00JGL 6419753 IC50 = 4154 nM T65864 D00NWF 5730 IC50 = 180 nM T65864 D00PPB 11703439 IC50 = 450 nM T65864 D00TBD 10461815 IC50 > 10000 nM T65864 D00XOQ 9885504 IC50 = 1300 nM T65864 D01YWE 25207521 IC50 > 50000 nM T65864 D02NKV 5172 IC50 = 25 nM T65864 D03MUZ 17759555 IC50 = 11200 nM T65864 D04HWF 9871074 IC50 = 96 nM T65864 D05ZUX 44207909 Ki >= 1000 nM T65864 D06HVH 54613583 IC50 > 10000 nM T65864 D06LJL 9916282 IC50 > 100000 nM T65864 D06NUL 9819053 IC50 = 52 nM T65864 D07ADX 54764565 IC50 = 12050 nM T65864 D07IHM 9823787 IC50 > 10000 nM T65864 D07TTR 46886448 IC50 = 1260 nM T65864 D08BIP 64796 IC50 = 0.74 nM T65864 D08DSJ 9845197 IC50 = 4000 nM T65864 D08HFG 24809764 IC50 > 10000 nM T65864 D08LYB 5166 IC50 = 34 nM T65864 D08WFC 15311937 IC50 = 570 nM T65864 D09DRF 90334 IC50 = 100000 nM T65864 D09HBZ 9795838 IC50 = 630 nM T65864 D09HVH 135566652 IC50 > 10 nM T65864 D09HXU 16086113 IC50 = 3903 nM T65864 D09QBA 23378546 IC50 > 10000 nM T65864 D09XVY 7916852 IC50 = 1600 nM T65864 D0AY0F 70698427 IC50 > 10000 nM T65864 D0C3AD 10202642 IC50 = 7280 nM T65864 D0C7RS 1369 IC50 = 1200 nM T65864 D0E4LU 5171 IC50 = 160 nM T65864 D0E7VO 59627005 IC50 = 13.4 nM T65864 D0EW9J 10389239 IC50 > 100000 nM T65864 D0GD8Y 3006531 IC50 = 55000 nM T65864 D0GW4Q 5330524 IC50 = 50 nM T65864 D0H2PE 10236389 IC50 = 30 nM T65864 D0H6ZP 16654987 IC50 = 1030 nM T65864 D0H8RU 44405448 IC50 = 1400 nM T65864 D0J3LR 11634725 Ki > 4000 nM T65864 D0JR3W 71605047 IC50 = 43 nM T65864 D0K6YK 11676119 IC50 = 480 nM T65864 D0L0HG 766949 IC50 > 15848.93 nM T65864 D0M2OL 44404442 IC50 = 46 nM T65864 D0M3AR 5311276 IC50 = 1440 nM T65864 D0N9HX 44405454 IC50 = 600 nM T65864 D0OZ2S 11785878 IC50 > 10000 nM T65864 D0P3JW 447700 IC50 = 140 nM T65864 D0Q5UH 9858940 IC50 = 590 nM T65864 D0QN6U 9806182 IC50 = 2 nM T65864 D0QS9T 2352168 IC50 = 1500 nM T65864 D0S6GE 5327067 IC50 = 250 nM T65864 D0S9SX 11277481 IC50 = 15 nM T65864 D0T2RY 9948320 Ki >= 1000 nM T65864 D0V3OJ 6456587 IC50 = 1270 nM T65864 D0VC0I 5169 IC50 = 14.3 nM T65864 D0W4FF 6419739 IC50 = 380 nM T65864 D0X5CM 5289514 IC50 = 5 nM T65864 D0XB4P 447966 IC50 = 740 nM T65864 D0Y1SR 11844351 IC50 = 1300 nM T65864 D0ZG4G 11493598 Ki = 310 nM T65864 D0ZH1U 2051 IC50 = 560 nM T20333 D00STL 644241 IC50 = 677 nM T20333 D01PZD 5329098 IC50 = 84 nM T20333 D03ZBT 11626560 IC50 > 10000 nM T20333 D07NVU 9829523 IC50 = 142 nM T20333 D09KTS 24821094 IC50 > 1000 nM T20333 D0AZ3C 5291 IC50 = 960 nM T20333 D0E6XR 3062316 IC50 = 5.012 nM T20333 D0G6QF 3081361 IC50 = 1600 nM T20333 D0R0MW 5329102 IC50 = 35 nM T20333 D0V9WF 126565 IC50 = 31 nM T20333 D0W5HK 216239 IC50 = 19 nM T20333 D00RYA 16750271 IC50 = 69 nM T20333 D00UZR 5330286 IC50 > 10000 nM T20333 D05EXN 58298316 IC50 = 28 nM T20333 D08HOM 46207586 Ki = 3.162 nM T20333 D08NDE 46184986 IC50 = 1.2 nM T20333 D09TAB 25151352 IC50 = 12 nM T20333 D0C5JQ 25230468 IC50 = 3.2 nM T20333 D0E3TC 44259 IC50 = 1.14 nM T20333 D0FD6D 11751922 IC50 = 78 nM T20333 D0H9FR 118295624 IC50 = 8.1 nM T20333 D0M9QZ 11485656 IC50 = 3 nM T20333 D0O1IM 58298318 IC50 = 2000 nM T20333 D0S7HM 16041424 IC50 = 10 nM T20333 D0SG7B 49831257 IC50 = 489 nM T20333 D0T2ER 24767976 IC50 = 10 nM T20333 D08IMD 16755780 IC50 = 6 nM T20333 D0IT6Q 3038522 IC50 = 3430 nM T20333 D0T3ME 156422 IC50 > 30000 nM T20333 C6Y9CV 151193 IC50 = 1240 nM T20333 CL1M8I 350716 IC50 = 600 nM T20333 C10HLD 736073 IC50 > 10000 nM T20333 CA56NR 738703 IC50 = 1000 nM T20333 CX93VI 889132 IC50 = 4400 nM T20333 CHOQ59 953649 IC50 = 78 nM T20333 CLAZ82 2039872 IC50 = 390 nM T20333 CITV26 2724446 IC50 = 38 nM T20333 CHC5I0 2971839 IC50 > 10000 nM T20333 CFY1D0 2974957 IC50 > 10000 nM T20333 CFO6K8 2995620 IC50 = 47 nM T20333 C3BI5X 2996559 IC50 = 1900 nM T20333 CZB15R 4350438 IC50 = 4000 nM T20333 C5VW6K 5328016 IC50 > 20000 nM T20333 C5SF3R 6456015 IC50 = 12 nM T20333 CUPQ08 6539985 IC50 = 3 nM T20333 CMEZ23 6540005 IC50 = 57 nM T20333 C9TAL6 9826308 IC50 = 620 nM T20333 CX10KR 9828962 IC50 = 3430 nM T20333 C41QWA 9857146 IC50 > 10000 nM T20333 CW8V0K 9864418 IC50 > 20000 nM T20333 C1SV0B 9882621 IC50 = 500 nM T20333 CZCQ53 9884318 IC50 = 24 nM T20333 CHF7G5 9890746 IC50 > 30000 nM T20333 C3EUB4 9911005 IC50 > 30000 nM T20333 CLEC85 9945927 IC50 = 9 nM T20333 C37GXK 9983303 IC50 > 20000 nM T20333 C2C1BP 10089048 IC50 > 20000 nM T20333 CJQ68X 10108847 IC50 = 13 nM T20333 C7TA9J 10113568 IC50 = 38.9 nM T20333 CIV15Q 10113978 IC50 = 146 nM T20333 C5WCL2 10117540 IC50 = 5460 nM T20333 C0D1WF 10132097 IC50 = 33 nM T20333 C5RX9V 10155136 IC50 = 10 nM T20333 CD7J3O 10231458 IC50 = 1400 nM T20333 CC9E5Q 10249989 IC50 = 14000 nM T20333 C53QNY 10271800 IC50 = 6 nM T20333 C6F2SB 10271801 IC50 = 52 nM T20333 CG1AW8 10291931 IC50 = 15 nM T20333 CY6S4U 10292887 IC50 = 16 nM T20333 C95LYF 10457505 IC50 > 30000 nM T20333 CRX6F0 10479082 IC50 > 20000 nM T20333 CJ4P5T 10905857 IC50 > 30000 nM T20333 CW5C9X 11186250 IC50 = 1584.89 nM T20333 CDT27E 11186408 IC50 = 190 nM T20333 CO0I7K 11209405 IC50 = 120 nM T20333 CQ6B1N 11220125 IC50 = 47 nM T20333 CG9E2Y 11231718 IC50 = 36 nM T20333 CC4X1F 11232236 IC50 = 63 nM T20333 C0W9MS 11232263 IC50 > 10000 nM T20333 C49TGO 11232741 IC50 = 380 nM T20333 C5MEL1 11277266 IC50 = 400 nM T20333 CJ4Y3G 11280046 IC50 = 34 nM T20333 CM0IR4 11301179 IC50 = 1900 nM T20333 CQ54KI 11327103 IC50 = 37 nM T20333 C2AX3H 11328012 IC50 = 160 nM T20333 C64NDH 11336497 IC50 = 140 nM T20333 CST79V 11347784 IC50 = 360 nM T20333 CWN24F 11347957 IC50 = 550 nM T20333 C83YOL 11358866 IC50 = 280 nM T20333 C0J2TB 11359024 IC50 > 50000 nM T20333 C25ZCN 11374110 IC50 = 30 nM T20333 CM30TC 11387552 IC50 < 10 nM T20333 C4D6LW 11395681 IC50 = 80 nM T20333 CREQ51 11429654 IC50 = 27 nM T20333 CY0A4E 11429729 IC50 = 40 nM T20333 CJH2M5 11460725 IC50 = 1100 nM T20333 C3SOA0 11484747 IC50 = 130 nM T20333 CK3M0T 11495270 IC50 = 3 nM T20333 CL17QT 11497455 IC50 = 1.1 nM T20333 CI4J1W 11502118 IC50 = 80 nM T20333 CKXM76 11502358 IC50 = 940 nM T20333 CZ5Y8W 11502871 IC50 = 0.8 nM T20333 C97WGN 11505187 IC50 = 2.4 nM T20333 CV4W3K 11510315 IC50 = 1.3 nM T20333 C2T8YD 11511361 IC50 = 1.5 nM T20333 CP8B7T 11511719 IC50 = 3.8 nM T20333 CVNP35 11517292 IC50 = 2 nM T20333 CG3BZ9 11517980 IC50 = 100 nM T20333 C4GLJ5 11524843 IC50 = 1.4 nM T20333 CQ3TO7 11526741 IC50 = 1.8 nM T20333 C4Q8VK 11533340 IC50 = 1.3 nM T20333 CTG83F 11539329 Ki > 2500 nM T20333 C9SN0A 11545281 IC50 = 64 nM T20333 CD4LG5 11545419 IC50 = 28 nM T20333 CMF4T0 11545796 IC50 = 630 nM T20333 COY86F 11555179 IC50 = 0.4 nM T20333 CACS26 11561968 Ki > 2000 nM T20333 CD9SM0 11562361 IC50 = 1.6 nM T20333 CNZ10W 11567250 IC50 = 71 nM T20333 C8XBE5 11567957 IC50 = 16 nM T20333 CK8C1V 11568950 IC50 = 60 nM T20333 C30DKO 11574080 IC50 = 3 nM T20333 CTQU78 11574082 IC50 = 8 nM T20333 CE30QF 11574855 IC50 = 37 nM T20333 CC81KV 11575682 IC50 = 0.8 nM T20333 CTVX46 11576269 IC50 = 0.7 nM T20333 CU41YS 11577079 IC50 = 1.6 nM T20333 C3VUO7 11588815 IC50 = 2 nM T20333 CB91RQ 11589811 IC50 > 1000 nM T20333 CA2KX0 11590078 IC50 = 9 nM T20333 CM65QP 11590120 IC50 > 800 nM T20333 CMIL86 11590363 Ki > 2500 nM T20333 C12PEW 11592380 IC50 = 0.83 nM T20333 CKJ4G0 11606814 IC50 = 1.1 nM T20333 C97NOU 11606951 IC50 = 1 nM T20333 CQYD09 11610817 IC50 = 18 nM T20333 CF5G9P 11611808 IC50 = 0.7 nM T20333 C6LUG4 11612700 IC50 = 2.7 nM T20333 CXM3C2 11619776 IC50 = 0.9 nM T20333 C5B3XJ 11620410 IC50 = 80 nM T20333 C4WB8P 11621465 IC50 = 0.3 nM T20333 CST9A4 11625534 IC50 = 25 nM T20333 CSM62L 11626920 IC50 = 5 nM T20333 C3CP2G 11627368 IC50 = 1.3 nM T20333 C7CG3P 11627369 IC50 = 2.5 nM T20333 C7W3TE 11633427 IC50 > 1000 nM T20333 CYL45U 11634544 IC50 = 1.1 nM T20333 C52ZKM 11634651 IC50 = 2.6 nM T20333 C5TJ0U 11640458 IC50 = 60 nM T20333 C9T6SC 11640926 Ki > 2500 nM T20333 CTXG50 11642625 IC50 = 22 nM T20333 CP91IG 11642786 IC50 = 0.62 nM T20333 CZPG34 11650178 IC50 = 1.7 nM T20333 CQ4OC2 11654378 IC50 = 0.78 nM T20333 CWU8T0 11654827 IC50 = 0.7 nM T20333 CKB27X 11661133 IC50 = 60 nM T20333 C87BCA 11661428 IC50 = 470 nM T20333 CO15KF 11664409 IC50 = 1 nM T20333 CC7Q0S 11669846 IC50 = 0.8 nM T20333 CK4EB3 11682482 IC50 = 10 nM T20333 CBP2F7 11682855 IC50 = 890 nM T20333 C86AXS 11682945 IC50 = 10 nM T20333 CW3B2X 11685397 IC50 = 0.6 nM T20333 C10BSX 11689712 IC50 = 1.7 nM T20333 CD8VP2 11690004 IC50 = 1 nM T20333 CU0E8O 11690457 Ki > 2000 nM T20333 CH96LS 11692059 IC50 = 1.7 nM T20333 CI7OK8 11692969 IC50 = 10 nM T20333 CS6EG9 11695784 IC50 = 21 nM T20333 C3WCO9 11696478 IC50 = 1 nM T20333 CQ1PB6 11698112 IC50 = 83 nM T20333 CVL10S 11698924 IC50 = 1.4 nM T20333 C4DJ1V 11699804 IC50 = 1.3 nM T20333 CXZV40 11704205 IC50 = 720 nM T20333 CY97HJ 11710948 IC50 = 11 nM T20333 C32UEK 11718670 IC50 = 3.3 nM T20333 CUB2N6 11719537 IC50 = 600 nM T20333 CD9A0J 11720104 IC50 = 1.1 nM T20333 C9P0VD 11729539 IC50 > 30000 nM T20333 C8MOK3 11750699 IC50 < 1000 nM T20333 C8EB4Y 11775063 Ki = 5.012 nM T20333 CF45IM 15983970 IC50 = 5 nM T20333 CD9V0O 15983971 IC50 = 2300 nM T20333 CFPW41 16007116 Ki > 2500 nM T20333 CBL76D 16049231 IC50 = 1800 nM T20333 CNP38U 16049297 IC50 = 3300 nM T20333 CY31FX 16058788 IC50 = 1.2 nM T20333 C0D5NI 16058789 IC50 = 3.2 nM T20333 C7RO0W 16058790 IC50 = 8 nM T20333 C7FQ0H 16058898 IC50 = 35 nM T20333 CE8Z2O 16059012 IC50 = 22 nM T20333 C9JK2M 16059071 IC50 = 14 nM T20333 CD7EN8 16059072 IC50 = 21 nM T20333 CE30ZP 16059139 IC50 = 81 nM T20333 C5U4RC 16059142 IC50 = 420 nM T20333 CUA7N2 16059271 IC50 = 250 nM T20333 CG23AV 16059276 IC50 = 1100 nM T20333 CW6UJ9 16059338 IC50 = 13 nM T20333 CQ59OG 16059339 IC50 = 31 nM T20333 CF9QS8 16059340 IC50 = 68 nM T20333 C3Z4FP 16059404 IC50 = 730 nM T20333 CUL0E7 16059533 IC50 = 93 nM T20333 C0LQU6 16059534 IC50 = 8 nM T20333 C4M1DN 16059535 IC50 = 1.4 nM T20333 C89HSP 16059537 IC50 = 12 nM T20333 C3ZAK6 16059666 IC50 = 8 nM T20333 C63IGL 16059726 IC50 = 7 nM T20333 CH7MS6 16059729 IC50 = 0.8 nM T20333 CQG45C 16109001 IC50 = 25000 nM T20333 CGC34R 16118737 IC50 = 40 nM T20333 C5VPH9 16129448 IC50 = 9060 nM T20333 CP3HS4 16220354 IC50 = 8 nM T20333 CU56EW 16664858 IC50 > 10000 nM T20333 CK9IU2 16718491 IC50 = 1.2 nM T20333 C0V8FB 16730091 IC50 = 20 nM T20333 CA24TE 16730092 IC50 = 100 nM T20333 CDZ31W 16747696 IC50 = 45 nM T20333 CJ12TI 16755734 IC50 = 1.7 nM T20333 CU35QY 16755735 IC50 = 2.1 nM T20333 C35IWY 17938625 IC50 = 2000 nM T20333 C7ZK1E 17938633 IC50 = 500 nM T20333 CI62OL 18451141 Ki = 7.943 nM T20333 C8MQ2N 18770775 IC50 = 4000 nM T20333 CY97MC 18770784 IC50 = 1500 nM T20333 C1HCE3 18770799 IC50 = 5000 nM T20333 C72EWO 18770811 IC50 = 1600 nM T20333 C4BTV7 18770818 IC50 = 2100 nM T20333 C3JP7K 18770822 IC50 = 5000 nM T20333 C1GAJ2 18770840 IC50 > 100000 nM T20333 C5LUT8 22170188 IC50 = 29 nM T20333 C8B2VG 22170203 IC50 = 46 nM T20333 C3HN1W 22170205 IC50 = 18 nM T20333 CIB02C 22170247 IC50 = 22 nM T20333 CLY9S8 22170249 IC50 = 200 nM T20333 C9PZ1X 22170285 IC50 = 31 nM T20333 CH1O0G 22170297 IC50 = 36 nM T20333 CZC40B 22170298 IC50 = 100 nM T20333 C18NQU 22170305 IC50 = 18 nM T20333 CT5X0G 22170354 IC50 = 25 nM T20333 C1PR6W 22692676 IC50 > 50000 nM T20333 CIF8W2 23629682 IC50 = 4 nM T20333 CS16QD 23630085 IC50 = 3 nM T20333 CW7S4N 23630121 IC50 = 5 nM T20333 C9AN0Y 23630122 IC50 = 3 nM T20333 CZ12JX 23630124 IC50 = 10 nM T20333 C82TMH 23630125 IC50 = 4 nM T20333 C1RT4E 23630126 IC50 = 6 nM T20333 CD40IE 23630127 IC50 = 7 nM T20333 CQL7Y4 23630162 IC50 = 7 nM T20333 C07QDG 23630167 IC50 = 7 nM T20333 CI6C1R 23658582 IC50 = 71 nM T20333 C2RV3U 24180608 IC50 = 550 nM T20333 CHU49V 24757938 IC50 = 20 nM T20333 CRGK92 24758021 IC50 = 20 nM T20333 CLQ6K9 24758022 IC50 = 41 nM T20333 CNL96J 24758024 IC50 = 2 nM T20333 CTP5Y3 24758149 IC50 = 13 nM T20333 C02RHJ 24758150 IC50 = 3.7 nM T20333 CI5MQ9 24758151 IC50 = 23 nM T20333 CH1FR4 24758272 IC50 = 1.5 nM T20333 CD75UV 24758273 IC50 = 2.8 nM T20333 C4CKE6 24758274 IC50 = 1.4 nM T20333 C5TB4O 24758275 IC50 = 1.5 nM T20333 CID98M 24758276 IC50 = 1.4 nM T20333 CRI52D 24758277 IC50 = 7.1 nM T20333 C0D2PA 24758868 IC50 = 80 nM T20333 C3K5YO 24758982 IC50 = 700 nM T20333 CYU0Z8 24758983 IC50 = 500 nM T20333 CJL67N 24759089 IC50 = 200 nM T20333 C2APK8 24759090 IC50 = 500 nM T20333 C5CRF6 24759091 IC50 = 50 nM T20333 CA8U7X 24759094 IC50 = 100 nM T20333 C9W3SB 24759170 IC50 = 4.5 nM T20333 C3OY6A 24759171 IC50 = 4.5 nM T20333 C8TQ2R 24759173 IC50 = 11 nM T20333 CRB89L 24759205 IC50 = 30 nM T20333 CY7FG8 24759282 IC50 = 1.9 nM T20333 CZR43P 24759283 IC50 = 3.7 nM T20333 CBX56C 24759284 IC50 = 2.3 nM T20333 C9OM3V 24759285 IC50 = 6.8 nM T20333 CWQR59 24759286 IC50 = 4.6 nM T20333 C13JUP 24759314 IC50 > 1000 nM T20333 CVJA29 24759399 IC50 = 1.6 nM T20333 CH5Y7N 24759401 IC50 = 2.4 nM T20333 C50CYU 24759507 IC50 = 3.6 nM T20333 CE6Q7Y 24759508 IC50 = 2.2 nM T20333 CK6WB0 24759510 IC50 = 23 nM T20333 C7YG1N 24759534 IC50 = 41 nM T20333 CDF15M 24759558 IC50 < 3 nM T20333 CZHB78 24759614 IC50 > 60 nM T20333 CFOJ47 24759718 IC50 = 10 nM T20333 C7SO6V 24759719 IC50 = 1.9 nM T20333 C9Q3EW 24759721 IC50 = 6.9 nM T20333 CQNP54 24764449 IC50 = 238 nM T20333 C9FO8D 24783100 IC50 = 2.3 nM T20333 CU2KF4 24783102 IC50 = 0.5 nM T20333 CLFV60 24783104 IC50 = 0.4 nM T20333 CM7GH9 24783356 IC50 = 0.9 nM T20333 CN9HR4 24783357 IC50 = 0.3 nM T20333 CZM3X6 24783358 IC50 = 0.8 nM T20333 CXM08Q 24783618 IC50 = 2.9 nM T20333 C89ICH 24785380 IC50 = 1 nM T20333 C61KPI 24856363 IC50 > 20000 nM T20333 C12WLB 24874762 IC50 = 2.7 nM T20333 C8AGC3 24874798 IC50 = 5.9 nM T20333 CTE2D9 24874800 IC50 = 1.7 nM T20333 C8DPJ4 24874843 IC50 = 3.5 nM T20333 CR5Z9A 24874845 IC50 = 1.5 nM T20333 CNDQ53 24874846 IC50 = 7.2 nM T20333 CPDY61 24874883 IC50 = 0.6 nM T20333 C9Q0DK 24874884 IC50 = 2.1 nM T20333 C25LQE 24874885 IC50 = 0.9 nM T20333 CNHY40 24874886 IC50 = 2.3 nM T20333 CJ67CB 24874887 IC50 = 1.2 nM T20333 CR07FQ 24874972 IC50 = 13 nM T20333 CJ0CK5 24875075 IC50 = 1.4 nM T20333 C5BLF1 24875123 IC50 = 3.2 nM T20333 C49KUH 24875222 IC50 = 0.8 nM T20333 C79EZH 24875260 IC50 = 0.7 nM T20333 C8A9FN 24875261 IC50 = 1.5 nM T20333 C85CSJ 24875262 IC50 = 1.7 nM T20333 CJ2CB0 24875263 IC50 = 1.9 nM T20333 C4BJK8 24875264 IC50 = 1.2 nM T20333 C9B2TF 24880043 IC50 = 0.4 nM T20333 C5FD1A 24937369 IC50 = 0.7 nM T20333 CO85YQ 24937370 IC50 = 0.5 nM T20333 CL30OQ 24937495 IC50 = 0.5 nM T20333 CO86MX 24937497 IC50 = 0.7 nM T20333 C7T1XU 24937622 IC50 = 0.8 nM T20333 COIR04 24937746 IC50 = 0.5 nM T20333 CR52YA 24937877 IC50 = 1.3 nM T20333 CB85LQ 24938120 IC50 = 1.3 nM T20333 C0NRW6 24938241 IC50 = 4.1 nM T20333 C9YN2Q 24967131 IC50 > 10000 nM T20333 C3DI7Y 24995523 IC50 = 15 nM T20333 CAW4C2 25021199 IC50 = 8 nM T20333 C4KG0Y 25022599 IC50 = 2.5 nM T20333 C2ICS7 25065806 IC50 = 3 nM T20333 CMD8J5 25094492 IC50 > 1000 nM T20333 C1G5IO 25094493 IC50 = 88 nM T20333 COS3T6 25094494 IC50 > 1000 nM T20333 CH90KV 25097876 IC50 > 1000 nM T20333 C9L5ID 25098154 IC50 = 73 nM T20333 C1DYP9 25098155 IC50 > 1000 nM T20333 C9P1IU 25098159 IC50 > 1000 nM T20333 C53XHG 25098428 IC50 > 1000 nM T20333 CAO38V 25098429 IC50 = 499 nM T20333 C7FI3O 25098430 IC50 = 21 nM T20333 CMB52V 25098432 IC50 = 301 nM T20333 CYQ75I 25104233 IC50 = 0.5 nM T20333 COX75C 25163930 IC50 = 80 nM T20333 C4V6YM 25218446 IC50 = 857 nM T20333 C9EB7U 25218447 IC50 > 5000 nM T20333 CK9B3O 25218448 IC50 > 5000 nM T20333 CXEG38 25218449 IC50 > 5000 nM T20333 C9B7WJ 25218450 IC50 > 5000 nM T20333 C0DX7M 25218451 IC50 = 40 nM T20333 C9EH6C 25218452 IC50 = 15 nM T20333 CP93LC 25218453 IC50 = 5 nM T20333 C8BSR0 25218454 IC50 = 4 nM T20333 CSJ3B0 25218455 IC50 = 40 nM T20333 C09UXI 25218456 IC50 = 10 nM T20333 CHL85A 25218457 IC50 = 9 nM T20333 CAL54P 25218458 IC50 = 9 nM T20333 CZQ1D3 25218459 IC50 = 2 nM T20333 C34OKZ 25218460 IC50 = 2 nM T20333 CPL34H 25218461 IC50 = 2000 nM T20333 CT4WX3 25218462 IC50 = 5000 nM T20333 CLW2D7 25218463 IC50 = 5 nM T20333 CDWO68 25218464 IC50 > 5000 nM T20333 C9Q8BW 25218650 IC50 = 75 nM T20333 CI5TA9 25218651 IC50 = 15 nM T20333 C3VN4H 25218652 IC50 = 5.2 nM T20333 CDG62F 25218653 IC50 = 1.7 nM T20333 CN15CU 25218654 IC50 = 0.8 nM T20333 CV6M7S 25218655 IC50 = 2.4 nM T20333 C2TXC6 25218656 IC50 = 2.2 nM T20333 CFLX26 25218657 IC50 = 0.7 nM T20333 CA61LV 25218658 IC50 = 0.8 nM T20333 C48MHP 25218659 IC50 = 0.3 nM T20333 CPC8L4 25218660 IC50 = 0.4 nM T20333 CP42XG 25218662 IC50 = 0.4 nM T20333 CC1R7V 25218663 IC50 = 5 nM T20333 CV13ZM 28408236 IC50 = 17 nM T20333 C8B6TY 42628503 EC50 < 500 nM T20333 CO42DC 44138048 IC50 > 10000 nM T20333 CL65QV 44138049 IC50 > 10000 nM T20333 CM0BW2 44355543 IC50 > 50000 nM T20333 C0VSJ3 44355545 IC50 > 20000 nM T20333 CIV6A3 44355618 IC50 = 180 nM T20333 CYR4C8 44355673 IC50 = 180 nM T20333 CM24OQ 44355891 IC50 = 20000 nM T20333 CHL4V6 44355892 IC50 > 20000 nM T20333 CYV2D7 44368815 IC50 = 99 nM T20333 COPG94 44427519 IC50 > 10000 nM T20333 CGV37F 44440254 IC50 = 113 nM T20333 C5JUV3 44440256 IC50 = 1271 nM T20333 CFB56S 44440259 IC50 = 190 nM T20333 CEW9G2 44440261 IC50 = 2975 nM T20333 CIJ31H 44444451 IC50 = 16 nM T20333 CV3XL1 44444453 IC50 = 63 nM T20333 C0VQE9 44444455 IC50 = 100 nM T20333 CF2PA9 44444456 IC50 = 130 nM T20333 C1I7JG 44444458 IC50 = 63 nM T20333 CMIG81 44444459 IC50 = 630 nM T20333 C8RUQ6 44444461 IC50 = 32 nM T20333 C5WQ3J 44444463 IC50 = 80 nM T20333 CTX2Z1 44444464 IC50 = 50 nM T20333 C48SIT 44444466 IC50 = 40 nM T20333 C4OBH7 44444467 IC50 = 160 nM T20333 CABQ28 44444469 IC50 = 40 nM T20333 C52QPH 44444470 IC50 = 32 nM T20333 CCBP29 44444471 IC50 = 32 nM T20333 CI23VY 44444472 IC50 = 100 nM T20333 CEYM65 44444473 IC50 = 1000 nM T20333 CI2J9N 44444474 IC50 = 3200 nM T20333 CYRO82 44444475 IC50 = 320 nM T20333 CH5YS9 44444476 IC50 = 160 nM T20333 C5FQY4 44444477 IC50 = 250 nM T20333 CZI5P6 44444479 IC50 = 50 nM T20333 CMP05E 44444480 IC50 = 25 nM T20333 CW43XR 44444481 IC50 = 32 nM T20333 CIYK04 44444482 IC50 = 130 nM T20333 CW5YC2 44444484 IC50 > 10000 nM T20333 CVR0A9 44444486 IC50 = 16 nM T20333 C80VAT 44444489 IC50 > 10000 nM T20333 CYE5R3 44444491 IC50 > 10000 nM T20333 C6SA2K 44444494 IC50 > 10000 nM T20333 C4QB8G 44444496 IC50 > 10000 nM T20333 CZK35I 44444498 IC50 = 50 nM T20333 CL7VZ2 44444501 IC50 = 320 nM T20333 CH4E2K 44444503 IC50 = 160 nM T20333 C1YT2U 44444514 IC50 = 260 nM T20333 CJE81L 44444515 IC50 = 720 nM T20333 C8LX4K 44444518 IC50 = 5300 nM T20333 C25MKN 44444522 IC50 > 10000 nM T20333 CGP7U1 44444533 IC50 = 43 nM T20333 C6I1CY 44444535 IC50 > 10000 nM T20333 CD2LH3 44444538 IC50 = 40 nM T20333 CO5U7Q 44444539 IC50 = 80 nM T20333 CO48ZH 44444541 IC50 = 63 nM T20333 CE63TQ 44444543 IC50 = 100 nM T20333 C5N9UJ 44444544 IC50 = 32 nM T20333 CF78JA 44444545 IC50 = 25 nM T20333 CAG59S 44444546 IC50 = 50 nM T20333 CL52UP 44444547 IC50 = 200 nM T20333 CP2ZM1 44444548 IC50 = 16 nM T20333 CL4T8K 44444549 IC50 = 80 nM T20333 CFQT09 44444550 IC50 = 80 nM T20333 C4X5CN 44444551 IC50 = 16 nM T20333 C7NQ5D 44444552 IC50 = 63 nM T20333 CAE03O 44444553 IC50 = 200 nM T20333 CP6O3F 44444555 IC50 = 100 nM T20333 CX7IA6 44444579 IC50 > 10000 nM T20333 CJ81QK 44444583 IC50 > 10000 nM T20333 CYGZ93 44444584 IC50 > 10000 nM T20333 CMRU38 44444585 IC50 > 10000 nM T20333 CO3WZ2 44444586 IC50 > 10000 nM T20333 C7VHM5 44444587 IC50 > 10000 nM T20333 CNBD43 44444588 IC50 = 47 nM T20333 CW2SO8 44444589 IC50 = 17 nM T20333 C2L3DU 44444590 IC50 = 90 nM T20333 CF4YV3 44444591 IC50 = 200 nM T20333 C6SC3M 44444592 IC50 = 37 nM T20333 C2ITM0 44444593 IC50 > 2000 nM T20333 C7MXC9 44444594 IC50 = 19 nM T20333 CU10GN 44447253 IC50 = 17 nM T20333 C6DR3S 44447259 IC50 = 52 nM T20333 CQ53PN 44447263 IC50 = 6.3 nM T20333 C2CJ0L 44447265 IC50 > 60 nM T20333 C8W5YG 44447872 IC50 = 36 nM T20333 CWV5N3 44449418 IC50 = 16 nM T20333 C6AH2P 44449419 IC50 = 5 nM T20333 CO2Y7X 44449421 IC50 = 15 nM T20333 CC1NR4 44449453 IC50 = 2 nM T20333 CP08ZW 44449456 IC50 = 38 nM T20333 C8MJ3B 44449485 IC50 = 54 nM T20333 C2OD3E 44453169 IC50 = 3 nM T20333 CVA16K 44453170 IC50 = 4 nM T20333 CG8VS2 44453172 IC50 = 180 nM T20333 C6F7NI 44453297 IC50 = 280 nM T20333 C3FG1K 44453532 IC50 = 56 nM T20333 CFUI62 44453586 IC50 = 56 nM T20333 CLK0W7 44453682 IC50 = 2.1 nM T20333 C7WJO1 44453908 IC50 = 180 nM T20333 C6I1TW 44560803 IC50 = 4 nM T20333 CKN40Z 44561800 IC50 = 89 nM T20333 CNK3U9 44561837 IC50 = 32 nM T20333 C6J3SL 44561838 IC50 = 10 nM T20333 CW0SJ8 44561875 IC50 = 25 nM T20333 CHJW16 44561876 IC50 = 14 nM T20333 CBDS81 44561877 IC50 = 9 nM T20333 CQL30H 44561878 IC50 = 16 nM T20333 CT38LP 44561916 IC50 = 8 nM T20333 CJQ6X0 44561917 IC50 = 5 nM T20333 CT03OZ 44561918 IC50 = 3 nM T20333 C5XRO7 44561919 IC50 = 3 nM T20333 C65YGO 44561920 IC50 > 50000 nM T20333 C8L5BD 44562058 IC50 = 11 nM T20333 C16GLY 44562059 IC50 = 13 nM T20333 CZS7K0 44562060 IC50 = 31 nM T20333 CP0YZ1 44562061 IC50 = 140 nM T20333 C1LK7Z 44563832 IC50 = 7 nM T20333 CM8C3H 44570804 IC50 = 52 nM T20333 CR3UA6 44570850 IC50 = 38 nM T20333 CAWM71 44570851 IC50 = 30 nM T20333 C5G6RI 44570852 IC50 = 31 nM T20333 CQ4HU6 44570888 IC50 = 26 nM T20333 C95JRD 44570889 IC50 = 13 nM T20333 C9RTK6 44570928 IC50 = 28 nM T20333 CH1T3Y 44570971 IC50 = 9 nM T20333 CGU4F1 44570972 IC50 = 100 nM T20333 CJOR07 44571015 IC50 = 22 nM T20333 C8N4XB 44571016 IC50 = 12 nM T20333 C2PX1O 44571017 IC50 = 17 nM T20333 CI3JH9 44571018 IC50 = 18 nM T20333 CVHZ62 44571019 IC50 = 3 nM T20333 CFY7N8 44571020 IC50 = 2 nM T20333 CO9BF8 44571021 IC50 < 3 nM T20333 CS2ZU1 44571022 IC50 = 6 nM T20333 C9JP4V 44571098 IC50 = 10 nM T20333 C6Q2KH 44571099 IC50 = 17 nM T20333 C6X1CS 44571100 IC50 = 7 nM T20333 CP7A3V 44571101 IC50 = 80 nM T20333 CJ0C3M 44571102 IC50 = 129 nM T20333 C9OXK3 44571103 IC50 = 59 nM T20333 C1TW6O 44571104 IC50 = 8 nM T20333 CCV1G7 44571105 IC50 = 110 nM T20333 C5MZ3V 44571106 IC50 = 3 nM T20333 CY72WX 44571143 IC50 = 13 nM T20333 C1POA2 44571144 IC50 = 10 nM T20333 CL7TZ3 44571145 IC50 < 1 nM T20333 CYL29Q 44571146 IC50 = 7 nM T20333 C0ZUI5 44571147 IC50 = 54 nM T20333 CRA51M 44571148 IC50 = 24 nM T20333 CNS8W6 44571149 IC50 = 23 nM T20333 CZ4C9L 44571150 IC50 = 11 nM T20333 C1X7KR 44571187 IC50 = 3 nM T20333 C40PFR 44571188 IC50 = 15 nM T20333 C89FJC 44571189 IC50 = 3 nM T20333 CC1E9U 44571190 IC50 = 6 nM T20333 CVI0L8 44571221 IC50 = 7 nM T20333 CVCQ45 44571222 IC50 = 22 nM T20333 CF9HQ2 44571223 IC50 = 7 nM T20333 C75YGT 44571224 IC50 = 23 nM T20333 C7Q1VU 44580077 IC50 = 7000 nM T20333 CL90SE 44580358 IC50 = 90 nM T20333 CK1VE7 44580420 IC50 = 700 nM T20333 CH2R7X 44580449 IC50 = 100 nM T20333 C1VH0C 44580532 IC50 > 20000 nM T20333 CXC52J 44580649 IC50 = 600 nM T20333 CE32BQ 44580689 IC50 = 4 nM T20333 C8Z5AX 44580778 IC50 = 90 nM T20333 CY1A7W 44593407 IC50 = 6900 nM T20333 C3LZ6B 44593434 IC50 = 11 nM T20333 CY3HW5 46224684 IC50 = 9200 nM T20333 C7NUY3 46847552 IC50 > 1000 nM T20333 C8KFL5 46870016 IC50 = 143 nM T20333 CLS29B 46872626 IC50 > 10000 nM T20333 CL4BZ8 46880842 IC50 = 40 nM T20333 C3QF5H 46880843 IC50 = 57 nM T20333 C57YIV 46880881 IC50 = 345 nM T20333 CI8B6A 46880882 IC50 = 1700 nM T20333 CFZL37 46880883 IC50 = 1990 nM T20333 CZM46J 46880884 IC50 = 56 nM T20333 CO4JM7 46880930 IC50 = 30 nM T20333 C98QZF 46880931 IC50 = 12 nM T20333 C2O8RZ 46886323 IC50 > 1000 nM T20333 CQLT07 46913878 IC50 < 1000 nM T20333 C60GAV 46929544 IC50 = 1580 nM T20333 CC8B0L 49798465 IC50 = 2.3 nM T20333 CJZH84 49798631 IC50 = 2.5 nM T20333 C3VEK4 49798632 IC50 = 1.9 nM T20333 C73PSQ 49805872 IC50 = 15 nM T20333 CML8Z5 49805873 IC50 = 8.9 nM T20333 C45LKE 49805998 IC50 = 13 nM T20333 CYG8Z4 49805999 IC50 = 4.4 nM T20333 C2HK8O 49806001 IC50 = 17 nM T20333 CMN0Y6 49806002 IC50 = 20 nM T20333 CEF9Q0 49806125 IC50 = 17 nM T20333 C41TPM 49806128 IC50 = 10 nM T20333 C64IXV 49806253 IC50 = 15 nM T20333 CHSF07 49806372 IC50 = 14 nM T20333 CJ3SU6 49830359 Ki = 1.995 nM T20333 CBCF39 49830372 Ki = 5.012 nM T20333 C8NA4L 53384644 IC50 > 30000 nM T20333 CO6B0E 54583043 IC50 > 10000 nM T20333 C3PGE2 54585958 IC50 > 10000 nM T20333 CV7HJ8 54585959 IC50 > 10000 nM T20333 C8AB1J 54759606 Ki = 230 nM T20333 CBO2L1 54761157 IC50 = 6.9 nM T20333 CS23GM 54762055 IC50 = 15 nM T20333 C9DX3J 56649281 IC50 = 10 nM T20333 C4WE9B 57391179 IC50 > 1000 nM T20333 CY10TP 57391180 IC50 = 600 nM T20333 CU3DM9 57391295 IC50 > 1000 nM T20333 CU7J9C 57393063 IC50 = 90 nM T20333 CD4HS3 57393074 IC50 > 1000 nM T20333 CS60KL 57393075 IC50 > 1000 nM T20333 CKVG97 57394105 IC50 < 1000 nM T20333 CWMT98 57394785 IC50 > 1000 nM T20333 C9PY4Q 57394798 IC50 > 1000 nM T20333 C3F9VS 57394799 IC50 > 1000 nM T20333 C4CN6V 57396453 IC50 > 900 nM T20333 CCT58R 57396454 IC50 > 1000 nM T20333 CXA5Z9 57396541 IC50 = 40 nM T20333 CPAH35 57396542 IC50 = 200 nM T20333 CY8U1Q 57396557 IC50 = 300 nM T20333 C4J6UZ 57397845 IC50 < 1000 nM T20333 CWV96N 57398329 IC50 = 20 nM T20333 C8K1WJ 57398330 IC50 = 8 nM T20333 CBK02S 57399984 IC50 = 30 nM T20333 CNU4I7 57399985 IC50 = 100 nM T20333 CD9KF3 57399986 IC50 = 50 nM T20333 C0BA7P 57401686 IC50 > 1000 nM T20333 CH56JP 57401785 IC50 = 400 nM T20333 C7YMG1 57401804 IC50 > 1000 nM T20333 C20ZAX 57401805 IC50 = 30 nM T20333 C15YQW 57401806 IC50 = 300 nM T20333 CY5TJ9 57401807 IC50 > 600 nM T20333 C4L0SA 57401808 IC50 = 40 nM T20333 C4J0OD 57403506 IC50 = 10 nM T20333 CN0M3Z 57403518 IC50 > 1000 nM T20333 CZSM95 57412684 IC50 = 2800 nM T20333 C93PNS 57725464 IC50 = 2 nM T20333 CI50KU 58167984 IC50 = 575 nM T20333 CU3WG8 58298312 IC50 = 2700 nM T20333 CHAB28 58994325 IC50 = 8 nM T20333 CSP3L0 58994366 IC50 = 19 nM T20333 CD2WR4 58994369 IC50 = 0.7 nM T20333 CK52WC 58994383 IC50 = 2 nM T20333 C9Q8AW 58994385 IC50 = 1.5 nM T20333 CASG36 58994416 IC50 = 2.4 nM T20333 CX6K1H 58994468 IC50 = 1.3 nM T20333 C6I0BA 58994487 IC50 = 3.5 nM T20333 C19ILC 58994517 IC50 = 0.6 nM T20333 C86KUI 58994523 IC50 = 3.5 nM T20333 CB8X9L 58994545 IC50 = 2 nM T20333 C43YRO 58994566 IC50 = 4.5 nM T20333 CP6Q7F 58994591 IC50 = 5.7 nM T20333 CK3LR6 58994593 IC50 = 0.8 nM T20333 CPJ1X6 59176320 IC50 > 1000 nM T20333 C3L4JY 59176329 IC50 = 767 nM T20333 CI8AL0 59176330 IC50 = 873 nM T20333 CDJQ62 59176336 IC50 > 1000 nM T20333 C2WXU1 59176348 IC50 = 312 nM T20333 CK68HX 59593266 IC50 = 62 nM T20333 CXJ63M 59603829 IC50 = 100 nM T20333 CQEU96 59603842 IC50 = 3.3 nM T20333 C78FOB 59633910 IC50 = 62 nM T20333 CPJQ50 59633916 IC50 = 86 nM T20333 CD6R5G 59633936 IC50 = 53 nM T20333 C0H2OQ 59633940 IC50 = 2216 nM T20333 CE28DO 59633994 IC50 = 12 nM T20333 C74TVO 59634010 IC50 = 12 nM T20333 CN9Q8I 59634020 IC50 = 11 nM T20333 CHR69F 59634027 IC50 = 13 nM T20333 CNF86I 59634031 IC50 = 12 nM T20333 CVT79N 59634040 IC50 = 25 nM T20333 C1ZY8J 59634050 IC50 = 41 nM T20333 CC14WX 59634061 IC50 = 9.1 nM T20333 CV3MN0 59634096 IC50 = 145 nM T20333 CWV4K6 59634103 IC50 = 29 nM T20333 CWFY29 59634114 IC50 = 64 nM T20333 CSA57R 59634115 IC50 = 15 nM T20333 C21UMF 59634122 IC50 = 18 nM T20333 C1MR8Q 60097495 IC50 > 1000 nM T20333 C51XCV 66781377 IC50 = 282 nM T20333 CF2Y0H 66781440 IC50 = 131 nM T20333 C1GJX2 66781520 IC50 = 384 nM T20333 C37NKO 67129970 IC50 > 10000 nM T20333 CK80LJ 67130050 IC50 > 10000 nM T20333 CV63UL 67240318 IC50 > 10000 nM T20333 C7GRV2 68755406 IC50 > 10000 nM T20333 C5DGR9 69036886 IC50 = 12 nM T20333 CCS20X 69063773 IC50 = 300 nM T20333 CH6S7Q 70681377 Ki = 3.162 nM T20333 CEB12M 70681395 IC50 = 200 nM T20333 CH27DE 70681409 IC50 = 100 nM T20333 CN29RI 70681410 IC50 = 100 nM T20333 CG93IE 70683519 IC50 = 10 nM T20333 CXSN14 70685622 IC50 > 900 nM T20333 CL24MP 70687766 IC50 = 20 nM T20333 C51DHN 70689791 IC50 = 500 nM T20333 C6ITV3 70689792 IC50 = 3 nM T20333 CMLY63 70689816 IC50 = 5 nM T20333 C08ASR 70689830 IC50 = 600 nM T20333 C4TF3G 70691955 IC50 = 600 nM T20333 CTWD94 70691956 IC50 > 1000 nM T20333 CIK5N2 70691957 IC50 = 300 nM T20333 C8RZP3 70691958 IC50 = 9 nM T20333 C0XRC9 70691981 IC50 = 200 nM T20333 C9RT8C 70693982 IC50 = 5 nM T20333 C2X1KJ 70694006 IC50 = 4 nM T20333 C54VLD 70694007 IC50 < 0.3 nM T20333 C6O3SM 70696108 IC50 > 1000 nM T20333 C48ZLN 71060894 IC50 < 40 nM T20333 C10CHQ 71060955 IC50 = 12 nM T20333 CWO0S3 71061505 IC50 = 17 nM T20333 CKT60L 71455860 Ki = 2100 nM T20333 CKNB62 71720020 IC50 = 22 nM T20333 CH91OY 72545066 IC50 = 5.6 nM T20333 C0JWR9 72545067 IC50 = 2.6 nM T20333 CCG6K8 72695028 IC50 = 12 nM T20333 C9OQ2I 72710839 IC50 = 1100 nM T20333 C6R8DI 72943374 IC50 = 2 nM T20333 C2B6QM 72943377 IC50 = 23 nM T20333 CI72LT 72943378 IC50 = 13 nM T20333 C7BJ4D 72943501 IC50 = 9 nM T20333 C2S6RL 72943502 IC50 = 37 nM T20333 CZ5NM9 72943503 IC50 = 30 nM T20333 C5GP0V 72943504 IC50 = 26 nM T20333 CKZ85O 72943506 IC50 = 13 nM T20333 C59QLH 72943630 IC50 = 6 nM T20333 C0FD9Q 72943753 IC50 = 19 nM T20333 C50OCA 72943755 IC50 = 9 nM T20333 CK70DB 72943756 IC50 = 12 nM T20333 C7MWK2 72943867 IC50 = 10 nM T20333 CGDB30 74538658 IC50 = 46 nM T20333 C1G4OV 76328399 IC50 > 1000 nM T20333 C0GQ8S 86291490 IC50 = 46 nM T20333 C98UIL 87421352 IC50 = 5.5 nM T20333 C1HW4B 89735655 IC50 = 22000 nM T20333 CQ2OB9 90292687 IC50 = 1220 nM T20333 CJQ5N6 91936970 IC50 = 57000 nM T20333 CU02NF 118559124 IC50 = 46 nM T20333 C08KEM 122179540 IC50 = 3400 nM T20333 C3AJ4C 122179546 IC50 > 10000 nM T20333 CG0RP7 122179547 IC50 = 2500 nM T20333 C1A0SQ 122179548 IC50 = 5300 nM T20333 C5B6QT 122189918 IC50 = 9.95 nM T20333 C53MKI 122189949 IC50 = 216 nM T20333 C4X7SD 122192466 IC50 = 43 nM T20333 CLM7K3 122604539 IC50 > 10000 nM T20333 C01JHI 122604566 IC50 > 10000 nM T20333 CC58IQ 127043948 IC50 = 133 nM T20333 C6OMB1 132204257 IC50 = 154 nM T20333 C6ROQ3 132546210 IC50 = 227 nM T20333 CJ04HZ 132585195 IC50 = 160 nM T20333 CIK38Q 134229735 IC50 = 3.73 nM T20333 C9FUK2 135151360 IC50 = 3162.28 nM T20333 CLCO61 135398510 IC50 = 1 nM T20333 C1VO5T 135405783 IC50 > 20000 nM T20333 CD87IX 135421239 IC50 > 5000 nM T20333 CIH4Y6 135430734 IC50 = 416 nM T20333 CH3OT0 135442635 IC50 = 340 nM T20333 C16XLU 135454992 IC50 > 12500 nM T20333 CCJ4K1 135457822 IC50 = 140 nM T20333 C0YU3M 135458175 IC50 = 2100 nM T20333 C90TYO 135471215 IC50 = 1000 nM T20333 C1C9TY 135483665 IC50 = 90 nM T20333 C7F4RC 135489124 IC50 = 830 nM T20333 C09CRJ 135489139 IC50 = 340 nM T20333 CTQ7H3 135497054 IC50 = 720 nM T20333 CGA9O6 135499847 IC50 = 300 nM T20333 C64EMD 135500075 IC50 > 12500 nM T20333 C5XL6P 135507511 IC50 = 22 nM T20333 CVZ08D 135509841 IC50 = 4300 nM T20333 CTU89G 135531166 IC50 = 250 nM T20333 C3WMY7 135531176 IC50 = 320 nM T20333 CMQ97S 135545383 IC50 = 220 nM T20333 C1XT0I 135875689 IC50 = 11 nM T20333 C72DQW 136018630 IC50 = 110 nM T20333 CGS27J 136018639 IC50 = 200 nM T20333 C9VX4A 136018642 IC50 = 90 nM T20333 CV5G1P 136018645 IC50 = 140 nM T20333 C1PN7I 136018651 IC50 = 170 nM T20333 C43ZWE 136018659 IC50 = 90 nM T20333 CZ40FX 136018664 IC50 = 240 nM T20333 CB64RK 136018669 IC50 > 5000 nM T20333 C94NUE 137333440 IC50 = 0.5 nM T20333 C90FJW 137365215 IC50 = 4.6 nM T20333 C7ZYL2 137365217 IC50 = 14 nM T20333 CRKO38 137365218 IC50 = 883 nM T20333 C6K5WV 137365221 IC50 = 8.6 nM T20333 C1QZH5 137365233 IC50 = 21 nM T20333 CH9WK1 137632228 IC50 = 180 nM T20333 CW2I0X 137632429 IC50 = 10.1 nM T20333 CX4BG3 137632686 IC50 = 28 nM T20333 CWO6X5 137632753 IC50 < 0.5 nM T20333 C1IRD9 137632976 IC50 = 5.8 nM T20333 CAW72M 137633292 IC50 = 31.9 nM T20333 CNX0F9 137634126 IC50 = 3 nM T20333 CI1E8V 137634241 IC50 > 10000 nM T20333 CV6W3A 137634751 IC50 = 20 nM T20333 C42PMG 137634834 IC50 = 180.7 nM T20333 C2DT0F 137634837 IC50 = 4.4 nM T20333 CS24ZE 137635122 IC50 = 30 nM T20333 C9MJB3 137635188 IC50 = 5.2 nM T20333 C18FSE 137635348 IC50 = 20.7 nM T20333 CLU61E 137635383 IC50 = 4 nM T20333 CZ3W9X 137636239 IC50 = 10 nM T20333 C8BDC7 137636863 IC50 = 20 nM T20333 CC1DK7 137636884 IC50 = 370 nM T20333 C0YD2I 137637558 IC50 = 41.2 nM T20333 CIPT52 137638089 IC50 = 30 nM T20333 CG09DY 137638779 IC50 = 5.1 nM T20333 C1CJL8 137639161 IC50 = 3.4 nM T20333 CBM75H 137639408 IC50 = 15.2 nM T20333 C0SVI6 137639489 IC50 > 10000 nM T20333 C6GQ7X 137640210 IC50 = 350 nM T20333 CO05XC 137641159 IC50 = 1.7 nM T20333 CC7NA3 137641695 IC50 = 5.6 nM T20333 CDF05B 137641797 IC50 = 30.4 nM T20333 CEX71A 137643024 IC50 = 151 nM T20333 CSJ4F0 137643599 IC50 = 6.8 nM T20333 C3X8JZ 137644493 IC50 = 1800 nM T20333 CQ08RW 137644617 IC50 = 16.4 nM T20333 CMA01W 137645075 IC50 = 10.3 nM T20333 C7Q0KP 137645669 IC50 = 2.1 nM T20333 CQJ45H 137645835 IC50 = 22.7 nM T20333 CN2J6Z 137646310 IC50 = 25.8 nM T20333 CHOF26 137646593 IC50 = 0.9 nM T20333 CDU7X6 137647023 IC50 = 20 nM T20333 CRI7W4 137647547 IC50 = 28.4 nM T20333 CU3FK9 137647695 IC50 = 40 nM T20333 C1MO6F 137647858 IC50 = 5.8 nM T20333 CB2S1Q 137647872 IC50 = 10 nM T20333 CDWM98 137648631 IC50 = 4.9 nM T20333 CA0DL1 137648651 IC50 = 630 nM T20333 C68MVW 137649573 IC50 = 25.9 nM T20333 CQ4R1I 137650454 IC50 = 4.7 nM T20333 C1A6ZV 137650580 IC50 = 6.5 nM T20333 C4N2VA 137650617 IC50 = 13.2 nM T20333 C12JHN 137650629 IC50 = 5.5 nM T20333 CO6DY4 137651084 IC50 = 20.2 nM T20333 CM2WA6 137651258 IC50 = 4.5 nM T20333 CBP7D8 137651768 IC50 = 17.1 nM T20333 C0GB7L 137651865 IC50 = 10.3 nM T20333 CEU20L 137652422 IC50 = 80 nM T20333 CJ6S9T 137652622 IC50 = 6.7 nM T20333 CDJ1E5 137652860 IC50 = 13.6 nM T20333 C28QUP 137652864 IC50 = 4701 nM T20333 C2BWK8 137654090 IC50 = 1 nM T20333 CUP85I 137654607 IC50 = 10 nM T20333 CHR5Y4 137655134 IC50 = 20.1 nM T20333 CF4BR6 137655863 IC50 = 7.2 nM T20333 CJ1AL4 137656216 IC50 = 2 nM T20333 CDU1V6 137656806 IC50 = 12 nM T20333 C02CKX 137656919 IC50 = 7.8 nM T20333 C3QY0B 137657045 IC50 = 32 nM T20333 CE2F4M 137657262 IC50 = 14.8 nM T20333 CWE31H 137657545 IC50 = 4.5 nM T20333 C2W5XI 137657580 IC50 = 30.6 nM T20333 CZP9J1 137658032 IC50 = 6.2 nM T20333 CS14VU 137658122 IC50 = 14.8 nM T20333 CKVU74 137659511 IC50 = 11700 nM T20333 C73CXG 137659722 IC50 = 5 nM T20333 CKL97P 137659725 IC50 = 20.9 nM T20333 C4U2GQ 137660913 IC50 = 230 nM T20333 CD03NK 137661226 IC50 = 9 nM T20333 CMSH35 137661302 IC50 = 7 nM T20333 CSOE96 137661336 IC50 = 18.1 nM T20333 C2EJB9 137661577 IC50 = 20.6 nM T20333 CUY09E 137662185 IC50 = 25.2 nM T20333 CIWG23 138393067 IC50 = 351 nM T20333 CN0X5D 138454787 IC50 = 247 nM T20333 C07EKN 138454794 IC50 = 14.2 nM T20333 C6AK0N 139030518 IC50 = 18 nM T20333 CDR27C 142717204 IC50 = 7 nM T20333 C4V1GH 145714280 IC50 = 12.59 nM T20333 CTUF34 145966712 IC50 = 581 nM T20333 C4OD9Q 145967187 IC50 > 1000 nM T20333 C5VWH3 145970734 IC50 = 277 nM T20333 CN7EF3 145996526 IC50 = 0.7 nM T20333 C43YLZ 155512202 IC50 = 28.5 nM T20333 C5CM7G 155513098 IC50 = 1.3 nM T20333 C2MD1Q 155513187 IC50 > 10000 nM T20333 CSC7H4 155513588 IC50 > 1000 nM T20333 CZY3P1 155515039 IC50 = 20.2 nM T20333 CI6H0B 155521051 IC50 = 7.2 nM T20333 C24HYD 155521063 IC50 = 10.8 nM T20333 CA24HS 155522641 IC50 = 1.4 nM T20333 C4RHY5 155523325 IC50 = 16.6 nM T20333 CWO2I9 155526782 IC50 = 3.5 nM T20333 CD2R9Z 155527646 IC50 = 6.5 nM T20333 C3KI2F 155527702 IC50 > 1000 nM T20333 CRGO31 155528777 Ki = 129 nM T20333 CM0UE1 155528948 IC50 = 1720 nM T20333 CK43VL 155529052 IC50 = 263 nM T20333 CABW80 155530129 IC50 = 25.1 nM T20333 C2ND9P 155530364 IC50 = 120 nM T20333 CS69CA 155532132 IC50 = 3.9 nM T20333 C51EKO 155532748 IC50 = 5.9 nM T20333 C9CO0H 155532831 IC50 = 4890 nM T20333 CE0XW9 155534632 IC50 = 430 nM T20333 C1OU9S 155536550 IC50 = 16.1 nM T20333 C3LC9I 155536820 IC50 = 50.12 nM T20333 CX37HC 155537699 IC50 = 23.4 nM T20333 C2Y0QK 155538640 IC50 = 160.3 nM T20333 CFSP46 155538687 IC50 > 1000 nM T20333 CN87GR 155539831 IC50 = 318 nM T20333 CFRW28 155539871 IC50 > 1000 nM T20333 CP25WZ 155539880 IC50 = 25.12 nM T20333 CRWB75 155541147 IC50 = 2.4 nM T20333 CH32PU 155542068 IC50 = 20 nM T20333 C79KOE 155542820 IC50 = 1290 nM T20333 CKOF06 155545262 IC50 = 6.5 nM T20333 CVK4G2 155547382 IC50 = 1.4 nM T20333 CU5L0W 155547861 IC50 = 510 nM T20333 C61TRK 155551323 IC50 = 1400 nM T20333 CG6E3V 155552422 IC50 > 3000 nM T20333 C7O9MV 155553758 IC50 > 3000 nM T20333 CK0G9U 155555603 IC50 = 9 nM T20333 C92JPH 155555824 IC50 = 2.6 nM T20333 C2V4OX 155556890 IC50 = 218.9 nM T20333 C2ZB4H 155560579 IC50 = 780 nM T20333 CX10VA 155561288 IC50 = 1100 nM T20333 CV9N1E 155561907 IC50 = 8.1 nM T20333 CZ6Q7P 155562074 IC50 > 1000 nM T20333 C7NW3X 155563124 IC50 = 5.5 nM T20333 CV80QU 155566736 IC50 = 4420 nM T20333 C5VO6Q 155567958 IC50 = 3 nM T20333 CZP47J 155568655 IC50 > 3000 nM T20333 D00HVA 11624601 Ki > 2500 nM T20333 D00WSN 2996093 IC50 = 1100 nM T20333 D07OXC 11650194 IC50 = 37 nM T20333 D0D6MH 11617559 IC50 = 60 nM T20333 D0EE6A 6398883 IC50 = 380 nM T20333 D0FH3M 18770833 IC50 = 500 nM T20333 D0L0HG 766949 IC50 > 10000 nM T20333 D0Q3NG 11715520 Ki > 2500 nM T20333 D0Q4EQ 16742063 IC50 = 622 nM T20333 D0R2WK 16038120 IC50 = 50.12 nM T20333 D0S7IE 11658882 Ki > 2500 nM T20333 D0UN9O 3385203 IC50 = 300 nM T20333 D0V4EX 54760053 IC50 = 10.5 nM T20333 D0Y4BL 11676971 IC50 = 0.69 nM T97749 CJ73BT 45486346 Ki > 10000 nM T97749 C9ETC4 45486354 Ki > 10000 nM T97749 CVPG40 45486356 Ki = 55 nM T97749 CSQ2K4 45486357 Ki = 1388 nM T97749 CJ2W9V 75593418 Ki = 1.7 nM T97749 C0ET8W 137630787 Ki = 0.36 nM T97749 D0A6FZ 75593419 Ki = 0.24 nM T97749 D0Y9PH 45486355 Ki = 312 nM T24373 CDX8Y1 648404 IC50 = 424 nM T24373 C6MC7E 651937 IC50 = 68 nM T24373 C6J8TO 655946 IC50 = 492 nM T24373 CSP71E 10086156 IC50 = 10000 nM T24373 CH0DS5 44291428 IC50 > 100000 nM T24373 C8DA4B 44291434 IC50 = 10000 nM T24373 CF8QI6 46867136 IC50 = 496 nM T24373 CAT57S 46867137 IC50 = 473 nM T24373 C7ULQ4 46867138 IC50 = 152 nM T24373 CH3YP2 46867139 IC50 = 300 nM T24373 C0KRG4 46867140 IC50 = 189 nM T24373 CME80U 76311375 IC50 = 10000 nM T45597 CU0E8O 11690457 Ki = 100 nM T45597 CHSF07 49806372 IC50 > 1000 nM T45597 CAZQ43 51003133 IC50 > 1000 nM T98642 D0E3TC 44259 IC50 = 83.9 nM T98642 CLS29B 46872626 IC50 > 10000 nM T98642 CV63UL 67240318 IC50 > 10000 nM T98642 C7A0VL 67448836 IC50 = 2.6 nM T98642 C5I7RB 68229183 IC50 = 23 nM T98642 CAKM96 92044487 IC50 = 10.69 nM T98642 CY4D8I 135566504 Ki = 316.1 nM T98642 CG3UZ1 135927974 Ki > 1000 nM T98642 CZ7EX0 136183413 IC50 > 30000 nM T98642 CAY48B 137796972 IC50 = 0.5 nM T98642 CK64IS 142445421 IC50 = 21 nM T98642 CJ6G2Q 155512128 IC50 = 335.7 nM T98642 CC7KH8 155513198 IC50 = 26.13 nM T98642 CNS8C4 155513486 IC50 = 1266 nM T98642 CC40LJ 155514352 IC50 = 2.71 nM T98642 CSI9G0 155515882 IC50 = 3013 nM T98642 CGHW08 155517160 IC50 = 63.83 nM T98642 CK3PJ7 155522075 IC50 = 44.89 nM T98642 C52GKR 155523141 IC50 = 6.44 nM T98642 CSP3B5 155523265 IC50 = 1.56 nM T98642 CF5N4L 155524573 IC50 = 20.88 nM T98642 CZ69OX 155524581 IC50 = 143.9 nM T98642 C3Y0OC 155526766 IC50 = 586.1 nM T98642 C43EFO 155526840 IC50 = 25.1 nM T98642 C0TXI4 155526872 IC50 > 10000 nM T98642 CSNB17 155532304 IC50 = 894.3 nM T98642 C2VTL9 155533905 IC50 = 19.06 nM T98642 CYHW45 155536207 IC50 = 61.41 nM T98642 CSZ4E8 155537204 IC50 = 977.5 nM T98642 CE85SU 155544622 IC50 = 2.94 nM T98642 CIL82B 155545007 IC50 = 5238 nM T98642 CU4HC9 155546697 IC50 = 65 nM T98642 CL9P8B 155547625 IC50 = 642.9 nM T98642 CG1IO8 155547851 IC50 = 721.4 nM T98642 COA9C3 155548719 IC50 = 1505 nM T98642 CDFQ73 155548750 IC50 = 5.44 nM T98642 CM6EH5 155549086 IC50 = 64.46 nM T98642 CL1IQ7 155555907 IC50 > 10000 nM T98642 CK8PS6 155555945 IC50 = 2663 nM T98642 CA3CQ9 155556653 IC50 = 142.5 nM T98642 COYX64 155559881 IC50 = 4.59 nM T98642 CHZX64 155559917 IC50 = 4790 nM T98642 C9LX2F 155561880 IC50 = 7055 nM T98642 CZ3RN1 155563559 IC50 = 6415 nM T98642 CMJ1K5 155565418 IC50 = 321.3 nM T98642 C26NAJ 155567560 IC50 = 2440 nM T98642 CJ5SE2 155568417 IC50 = 223.7 nM T98642 D00ERW 44444843 Ki = 5195 nM T98642 D0Y2WP 67448186 IC50 = 28 nM T86437 D03ZBT 11626560 IC50 = 563 nM T86437 D04LKS 25126798 Ki = 0.09 nM T86437 D04LVK 57379345 IC50 = 3730 nM T86437 D0EG1I 9926791 IC50 = 0.5 nM T86437 D0Y7IC 44205240 IC50 = 0.99 nM T86437 D00RYA 16750271 IC50 = 2700 nM T86437 D02TUL 118115473 IC50 = 1640 nM T86437 D03HUX 49792852 IC50 > 10000 nM T86437 D03LWG 53235510 IC50 > 10000 nM T86437 D04QWQ 59422203 IC50 = 13.2 nM T86437 D05PCM 78323835 IC50 = 29 nM T86437 D06EIC 57928403 IC50 = 3.9 nM T86437 D07EHV 44814409 IC50 > 10000 nM T86437 D07HPJ 11476171 IC50 > 10000 nM T86437 D07JAG 58557659 IC50 = 8 nM T86437 D0BI3N 44595079 IC50 = 12 nM T86437 D0D5ZJ 25062766 IC50 = 11 nM T86437 D0D8KQ 25127112 IC50 = 10 nM T86437 D0DK5X 135567296 IC50 = 2.2 nM T86437 D0DK8X 50922691 IC50 = 75 nM T86437 D0E3TC 44259 IC50 = 0.627 nM T86437 D0G8BM 16722836 IC50 = 100 nM T86437 D0O0LS 25141092 IC50 = 112 nM T86437 D0PN8H 46216796 IC50 = 1280 nM T86437 D0S1XX 134821691 IC50 = 1 nM T86437 D0SG7B 49831257 IC50 = 10 nM T86437 D0GZ7B 5328779 IC50 = 3380 nM T86437 C1BE5N 3799 IC50 = 19952.62 nM T86437 CU68FI 78893 Ki > 3500 nM T86437 CV7W4J 176406 IC50 = 39810.72 nM T86437 C6ZB4U 790291 Ki = 4600 nM T86437 CGQM48 869412 Ki = 2100 nM T86437 C0XL5P 951379 Ki > 3500 nM T86437 C7ZUW6 1246120 Ki = 3100 nM T86437 CI1B7L 1247281 Ki > 3500 nM T86437 CP6BI3 1481965 IC50 = 30000 nM T86437 C3F0GS 3120536 Ki = 2200 nM T86437 CD67OL 4250390 Ki > 3500 nM T86437 C6SNL5 4393251 Ki > 3500 nM T86437 CG9RD4 4448318 IC50 = 8530 nM T86437 CK6L3O 5121684 Ki > 3500 nM T86437 CYA76E 9798589 IC50 > 100000 nM T86437 CRZ5T7 9815801 IC50 > 10000 nM T86437 CO70CQ 10107882 IC50 = 290 nM T86437 CP28QI 10154513 IC50 > 10000 nM T86437 C35JMD 10269598 IC50 = 1550 nM T86437 C7SFI1 10296883 IC50 = 7300 nM T86437 CK2RY9 11164105 IC50 = 1480 nM T86437 C58YUH 11993785 IC50 = 47 nM T86437 C0Y7MG 12083227 IC50 = 1700 nM T86437 CZI64D 12083230 IC50 = 670 nM T86437 C75SGK 12997800 IC50 = 2 nM T86437 C0DUA7 15953425 IC50 = 14 nM T86437 C3JWA6 15953427 IC50 = 18 nM T86437 CWZM24 15953526 IC50 = 16 nM T86437 C1U8XW 16109036 IC50 = 1300 nM T86437 CSE35D 16739464 IC50 = 1800 nM T86437 C20OFQ 16739508 IC50 = 650 nM T86437 CCP56J 16739905 IC50 = 200 nM T86437 CQ64XI 16739921 IC50 = 390 nM T86437 CM3UF8 16739935 IC50 = 3200 nM T86437 CFEP56 16739948 IC50 = 170 nM T86437 C23KZR 16739951 IC50 > 10000 nM T86437 C9OQ1G 16750272 IC50 = 8000 nM T86437 CW2SY5 16750291 IC50 = 420 nM T86437 CIX7U2 16750304 IC50 = 3000 nM T86437 C6A3XS 16750306 IC50 = 1500 nM T86437 CB2TK1 16750327 IC50 = 1900 nM T86437 CH4O1C 16750328 IC50 > 10000 nM T86437 C90MJD 16750331 IC50 > 10000 nM T86437 C7JW2E 18008439 IC50 > 10000 nM T86437 C6UAZ0 20820292 IC50 = 230 nM T86437 C87BYV 22282847 IC50 > 10000 nM T86437 CJ5GR1 22282945 IC50 > 7140 nM T86437 C50FBN 22282953 IC50 > 10000 nM T86437 C16TAZ 22484511 IC50 = 720 nM T86437 CE7K3W 23532567 IC50 > 10000 nM T86437 CUY98W 23585560 IC50 = 39 nM T86437 CD0R9O 24699546 Ki > 3500 nM T86437 C7YG1N 24759534 IC50 = 2300 nM T86437 CAJ4T2 24762205 IC50 > 10000 nM T86437 CQNP54 24764449 IC50 = 25000 nM T86437 CRO97A 24798484 IC50 = 184 nM T86437 CFS2M7 24798487 IC50 = 142 nM T86437 CLBP72 24798571 IC50 = 70 nM T86437 CX1U4S 24800423 IC50 = 710 nM T86437 C4T0DG 24800602 IC50 = 8900 nM T86437 CH3ZG7 24800604 IC50 = 5300 nM T86437 CBA02Y 24800776 IC50 = 210 nM T86437 C3UFG1 24801129 IC50 = 47 nM T86437 CVR8S1 24801650 IC50 = 760 nM T86437 CWV98O 24899557 IC50 = 1000 nM T86437 C5S7XA 24958852 IC50 = 58 nM T86437 CJ68PR 24958855 IC50 = 180 nM T86437 C0JYA9 25123154 IC50 = 390 nM T86437 C56JVD 25123155 IC50 = 91 nM T86437 CZM6Q2 25123472 IC50 = 35 nM T86437 C3IA7V 25123474 IC50 = 1500 nM T86437 C6V4NB 25123475 IC50 = 460 nM T86437 CFK89A 25123806 IC50 = 98 nM T86437 C3RMN9 25123807 IC50 = 250 nM T86437 C5GO3T 25123808 IC50 = 1850 nM T86437 C4WFL0 25128110 IC50 = 130 nM T86437 COV8Z0 25143021 IC50 > 10000 nM T86437 CI0E2L 25154395 IC50 = 970 nM T86437 CL1W5D 25154436 IC50 = 390 nM T86437 C0ZXH7 25236808 Ki = 1700 nM T86437 CT7X8Y 27700054 Ki > 3500 nM T86437 C9M1PO 42599880 IC50 = 547 nM T86437 C93PID 42599883 IC50 > 10000 nM T86437 CB9DS2 42600632 IC50 = 975 nM T86437 CIA57B 42600635 IC50 = 27 nM T86437 CH10ZY 42600886 IC50 > 10000 nM T86437 C3IT9C 42600887 IC50 > 4000 nM T86437 CY4LG8 42622934 IC50 = 1.5 nM T86437 CCB1E9 44124695 IC50 > 100000 nM T86437 CIT2A7 44192904 IC50 = 256.7 nM T86437 C3VRO9 44557921 IC50 = 4365.16 nM T86437 C5YL2S 44570390 IC50 = 490 nM T86437 C7DW0O 44602589 IC50 = 2.8 nM T86437 C6QT0J 44622837 IC50 > 1000 nM T86437 C4EBH7 44625519 IC50 > 4000 nM T86437 C02RNS 44625983 IC50 = 103 nM T86437 CKUA84 44626045 IC50 = 92 nM T86437 C7E1DT 44626178 IC50 = 23 nM T86437 C2SLI6 44631938 IC50 = 10 nM T86437 CU3RF1 45139989 IC50 > 10000 nM T86437 CQGZ06 45139991 IC50 > 10000 nM T86437 CZ7T8F 45275363 IC50 = 16 nM T86437 CB58EO 45275368 IC50 = 24 nM T86437 CU3AD0 45275473 IC50 = 28 nM T86437 CQ3KO2 45375955 IC50 = 58 nM T86437 CE45XW 46208354 IC50 = 2.9 nM T86437 CUHB49 46208355 IC50 = 2.5 nM T86437 CW38GO 46208357 IC50 = 3.5 nM T86437 C43COY 46208358 IC50 = 5.4 nM T86437 CE4Q7D 46208596 IC50 = 6.7 nM T86437 CM9UN7 46208601 IC50 = 0.24 nM T86437 CH7JB4 46209051 IC50 = 4.2 nM T86437 C7ON5A 46233287 IC50 > 10000 nM T86437 CWN3M0 46234565 IC50 = 92 nM T86437 CLTU68 46234566 IC50 = 26 nM T86437 C5YH1F 46235625 IC50 = 59 nM T86437 CC25DT 46235942 IC50 = 30 nM T86437 CZ7J6K 46236109 IC50 = 83 nM T86437 C1S4LH 46398810 IC50 = 303 nM T86437 C35AIH 46865430 IC50 = 48 nM T86437 C2EK4B 46865431 IC50 = 140 nM T86437 CMZ0R3 46865529 IC50 = 28 nM T86437 C3B2NL 46865530 IC50 = 82 nM T86437 CC2O9R 46865656 IC50 = 1584.89 nM T86437 CJ3NV8 46865657 IC50 = 130 nM T86437 C5NZ8R 46880686 IC50 = 680 nM T86437 CZ79VE 46880687 IC50 = 27.5 nM T86437 C0YNH6 46880737 IC50 = 22 nM T86437 CGO7C5 46880738 IC50 = 82 nM T86437 C75ZTG 46880739 IC50 = 180 nM T86437 C9T7WL 46880784 IC50 = 67 nM T86437 CSV4G2 46880785 IC50 = 35 nM T86437 C9MW2L 46885052 IC50 > 10000 nM T86437 C69HUW 46885053 IC50 = 940 nM T86437 CASL67 46885231 IC50 = 1200 nM T86437 CEU6O4 46885232 IC50 = 4700 nM T86437 CE27LI 46885233 IC50 = 89 nM T86437 CB8LN4 46885234 IC50 = 362 nM T86437 CMX7U6 46885289 IC50 = 190 nM T86437 CB1ZN5 46885290 IC50 = 60 nM T86437 C2B5XF 49765254 IC50 > 10000 nM T86437 CT7EY8 49817363 IC50 = 253 nM T86437 CMKB24 49838268 IC50 = 22 nM T86437 CB34CO 49839441 Ki = 360 nM T86437 C2DGY0 49839445 Ki > 3500 nM T86437 C06MKW 49839561 Ki = 83.8 nM T86437 CJZ5A0 49840306 IC50 > 10000 nM T86437 CF91RS 49843531 IC50 > 10000 nM T86437 C7A6IZ 49850211 IC50 = 20 nM T86437 C9UZ6E 49855558 IC50 > 10000 nM T86437 CR6Q5Y 49855559 IC50 = 1760 nM T86437 CTM0I6 49855750 IC50 = 1200 nM T86437 CJXR91 49855751 IC50 = 2240 nM T86437 C57FQH 49856318 IC50 = 2780 nM T86437 C70QSD 49856319 IC50 = 1120 nM T86437 C24SMN 49856320 IC50 > 10000 nM T86437 CHK7D3 49856321 IC50 = 840 nM T86437 C90VXM 49856700 IC50 = 1910 nM T86437 CK4LJ5 49856703 Ki = 610 nM T86437 CK5TH3 50906783 IC50 = 10 nM T86437 CA0WR3 50914031 IC50 = 170 nM T86437 CQE9D1 50925411 IC50 = 311 nM T86437 C2Y6QS 50938552 IC50 > 10000 nM T86437 CF26MU 50991562 IC50 = 6000 nM T86437 C20VEP 50994284 IC50 > 10000 nM T86437 CI1L0M 50994285 IC50 = 737 nM T86437 C7ZWT8 50994286 IC50 = 4700 nM T86437 C6VNE1 50994366 IC50 = 754 nM T86437 CSEZ73 50994367 IC50 = 6500 nM T86437 C1R8ZI 50995341 IC50 = 509 nM T86437 C53NRD 50995522 IC50 = 621 nM T86437 C9NYP4 51036677 IC50 > 10000 nM T86437 C4WRY3 51037112 IC50 > 10000 nM T86437 CRI28Z 51037948 IC50 > 10000 nM T86437 CA9DE6 52941228 IC50 = 500 nM T86437 C1T5EH 52942437 IC50 = 610 nM T86437 CEPS91 52943663 IC50 = 39 nM T86437 C2IQ5B 52943672 IC50 >= 10000 nM T86437 CTN0C3 52944839 IC50 = 990 nM T86437 CT2U3E 52947304 IC50 = 19 nM T86437 CQY9D0 52948526 IC50 = 45 nM T86437 C8TC3P 52948550 IC50 = 80 nM T86437 CIM43G 52948562 IC50 = 160 nM T86437 CL14DA 53317826 IC50 = 490 nM T86437 C72DMQ 53320251 IC50 > 7500 nM T86437 C2W9OA 53324451 IC50 > 10000 nM T86437 C0PLX8 53340959 Ki = 2.9 nM T86437 CN70RK 53341007 Ki = 9.1 nM T86437 CQS1R8 53341008 Ki = 16 nM T86437 CKS8G7 53341054 Ki = 9.3 nM T86437 CSUN84 53341057 Ki = 14 nM T86437 C4R2SW 53341104 Ki = 2.6 nM T86437 C4BM5W 53341107 Ki = 6.2 nM T86437 CZKQ72 53341161 Ki = 7.9 nM T86437 CN59SH 53341248 Ki = 2.4 nM T86437 CB83XH 53341368 Ki = 24 nM T86437 CD2CH6 53341413 Ki = 25 nM T86437 CGP23R 53341457 Ki = 0.4 nM T86437 CK7O6Y 53341461 Ki = 16 nM T86437 C9QEA5 53341463 Ki = 1.7 nM T86437 C7U1KW 53341498 Ki = 4.6 nM T86437 C5ZI7P 53341503 Ki = 0.9 nM T86437 C2MAO8 53341544 Ki = 22 nM T86437 C56TYK 53385837 IC50 = 430.5 nM T86437 CNLM53 53385838 IC50 = 361 nM T86437 C1XE2K 53385938 IC50 = 870.7 nM T86437 C37JTE 53385939 IC50 = 47 nM T86437 CV92IB 53386254 IC50 = 23 nM T86437 CU6QF7 53386309 IC50 < 0.5 nM T86437 CYU0R4 53386418 IC50 = 0.59 nM T86437 C7RM6Q 53386421 IC50 = 0.47 nM T86437 CEN91X 53389820 IC50 = 636.6 nM T86437 C37PHN 53497571 IC50 = 211 nM T86437 CCF1B3 53497572 IC50 = 1090 nM T86437 CY5C8A 54589404 IC50 = 3.2 nM T86437 CS7E0A 54672927 IC50 = 224.3 nM T86437 CHZ27O 54673255 IC50 = 24 nM T86437 C7X5ZM 54673258 IC50 = 75.8 nM T86437 CZ84NW 54673259 IC50 = 44.5 nM T86437 CX0U2A 54673422 IC50 = 44.8 nM T86437 C19FZK 54673425 IC50 = 1102.5 nM T86437 CBPT15 54673763 IC50 = 6300 nM T86437 C36BAI 54673911 IC50 = 108.1 nM T86437 CD8ZK6 54674056 IC50 = 220 nM T86437 CFTE97 54674369 IC50 = 840 nM T86437 CUCI05 54674990 IC50 = 99.7 nM T86437 CH0IM9 54754557 IC50 = 54 nM T86437 C1XS2J 54760383 IC50 = 3300 nM T86437 CXH2P4 54766274 IC50 = 370 nM T86437 CD28VZ 54766423 IC50 > 10000 nM T86437 CAP1J7 54766425 IC50 > 10000 nM T86437 C75JFM 54766426 IC50 > 10000 nM T86437 CDIC43 54766427 IC50 = 850 nM T86437 C2XDG1 54766428 IC50 = 5400 nM T86437 C0XCY1 54766576 IC50 = 2100 nM T86437 CPH3Y7 54766578 IC50 > 10000 nM T86437 C0T4SL 54766726 IC50 = 480 nM T86437 CZD70Q 54767039 IC50 = 74 nM T86437 CN1DZ6 54767189 IC50 = 150 nM T86437 C1W3EZ 56591424 IC50 = 3.5 nM T86437 CTB63S 56591428 IC50 = 79 nM T86437 CWR1P6 56591446 IC50 = 18 nM T86437 C6ZL7H 56592816 IC50 = 1200 nM T86437 C6Z1QA 56592817 IC50 = 24 nM T86437 CM8JX1 56604907 IC50 = 10000 nM T86437 CR9A5O 56834874 IC50 = 708 nM T86437 C58MSV 56834889 IC50 = 177 nM T86437 CBFR12 56925356 IC50 = 133 nM T86437 C80DRA 56925357 IC50 = 406 nM T86437 C0HUN8 56925358 IC50 = 307 nM T86437 C6Z2EA 56925359 IC50 = 8820 nM T86437 CC1MN2 56925454 IC50 = 3100 nM T86437 C3XC0T 56925455 IC50 = 377 nM T86437 CBW6T3 56925456 IC50 = 39 nM T86437 C8G3NO 56925457 IC50 = 70 nM T86437 CHS19C 56925458 IC50 = 36 nM T86437 CBMO42 56925459 IC50 = 78 nM T86437 CQTD41 56925550 IC50 = 129 nM T86437 CI9T3S 56925551 IC50 = 654 nM T86437 CS84ZU 56925552 IC50 = 206 nM T86437 C9IVD0 56929216 Ki = 1.8 nM T86437 CQ2F3C 56973424 Ki = 1.7 nM T86437 CSO40C 56973425 Ki = 2.4 nM T86437 CU5BD9 57336812 IC50 = 81 nM T86437 C31LJU 57339437 Ki = 10 nM T86437 CMF7J0 57339438 Ki = 45 nM T86437 CPO2J4 57342178 IC50 = 4800 nM T86437 CA93PN 57342180 IC50 = 5100 nM T86437 C9Z6QJ 57502388 IC50 = 43 nM T86437 COU4M1 57915982 IC50 = 20 nM T86437 C1G5SK 57916044 IC50 = 30 nM T86437 C3C0PQ 57916049 IC50 = 79 nM T86437 CH6RB0 57916164 IC50 = 24 nM T86437 C9MF8U 57928260 IC50 = 19 nM T86437 C3KQJ8 57928435 IC50 = 3.9 nM T86437 C5H8VE 57928583 IC50 = 12 nM T86437 C13VIO 57928632 IC50 = 110 nM T86437 C8BTO7 57928826 IC50 = 7.8 nM T86437 C8R4FE 57991377 IC50 = 134.3 nM T86437 CD6ZP3 58009815 EC50 = 430 nM T86437 CWU1Y3 58009825 EC50 = 1200 nM T86437 C8S6MY 58010054 IC50 = 3 nM T86437 CM1B4V 58010265 EC50 = 150 nM T86437 CQND09 58177229 IC50 = 231 nM T86437 CU4I8X 58177247 IC50 = 53 nM T86437 CLEH36 58177279 IC50 = 287 nM T86437 CIK3U8 58177332 IC50 = 129 nM T86437 C8D2TA 58177362 IC50 = 199 nM T86437 CYC85B 58177456 IC50 = 15 nM T86437 C7BU0H 58180518 IC50 = 22 nM T86437 CKA28H 58180521 IC50 = 16 nM T86437 C2I5LO 58180525 IC50 = 61 nM T86437 CN4OZ8 58180573 IC50 = 250 nM T86437 C92FOB 58180591 IC50 = 19 nM T86437 CWXC70 58180596 IC50 = 270 nM T86437 C9N1QB 58180623 IC50 = 330 nM T86437 CSK1U8 58180628 IC50 = 40 nM T86437 C6LT9S 58180630 IC50 = 46 nM T86437 CCBT87 58180639 IC50 = 40 nM T86437 C3MK9V 58374721 IC50 = 1.4 nM T86437 C7Q8YZ 58374808 IC50 = 2749 nM T86437 CP81TW 58394456 Ki = 62 nM T86437 C4H3FY 58394522 Ki = 1.6 nM T86437 CM6SK2 58394565 Ki = 12 nM T86437 C8NFX5 58394608 Ki = 19 nM T86437 C6HPO3 58394632 Ki = 8.5 nM T86437 CBJ47W 58394678 Ki = 96 nM T86437 CC05OW 58394694 Ki = 32 nM T86437 CK71MA 58394722 Ki = 150 nM T86437 C6A8NR 58394745 Ki = 1.2 nM T86437 CH4F5Y 58394751 Ki = 2 nM T86437 C0F3BO 58394783 Ki = 2.8 nM T86437 CLA74K 58394787 Ki = 4.9 nM T86437 C0Y6FH 58394796 Ki = 68 nM T86437 CO5TH6 58394820 Ki = 88 nM T86437 CY0UV6 58394828 Ki = 1.3 nM T86437 C0X7IK 58394837 Ki = 0.9 nM T86437 CW7D0O 58394866 Ki = 0.8 nM T86437 C0W2AT 58394878 Ki = 210 nM T86437 C97QAK 58394904 Ki = 5.8 nM T86437 C9Q4WD 58394916 Ki = 15 nM T86437 CI37CQ 58394927 Ki = 1.3 nM T86437 CFQW46 58394944 Ki = 2.9 nM T86437 C5RGU7 58394946 Ki = 121 nM T86437 CDP7J2 58394959 Ki = 4.3 nM T86437 CF8G9P 58394966 Ki = 50 nM T86437 C6KO0G 58395044 IC50 = 30 nM T86437 CASI81 58395078 Ki = 0.1 nM T86437 C2H4NS 58395107 Ki = 3.7 nM T86437 C3Y6WA 58395132 Ki = 9.3 nM T86437 CCK96S 58395150 Ki = 2.7 nM T86437 CTF2Z1 58395158 Ki = 2.6 nM T86437 C0GSU3 58395193 Ki = 13 nM T86437 CDK5L1 58395223 Ki = 1.5 nM T86437 CU04YA 58395228 Ki = 8.7 nM T86437 CWOB94 58395230 Ki = 0.6 nM T86437 C9J5UV 58395232 Ki = 2 nM T86437 CO7G2W 58395250 Ki = 7.3 nM T86437 C21OFZ 58395252 Ki = 8.3 nM T86437 CYC87B 58395253 Ki = 156 nM T86437 CQP86B 58395268 Ki = 28 nM T86437 CI7KN3 58395278 Ki = 5.8 nM T86437 CTX12W 58395280 Ki = 11 nM T86437 CWBM72 58395283 Ki = 0.3 nM T86437 CA8LU4 58395286 Ki = 5 nM T86437 C5S8BK 58395290 Ki = 18 nM T86437 CCHV76 58395300 Ki = 9.6 nM T86437 C4H2ZP 58395301 Ki = 1.1 nM T86437 CUS1M8 58395328 Ki = 43 nM T86437 C0WBQ9 58395366 Ki = 15 nM T86437 CWO4X6 58395380 Ki = 5.2 nM T86437 C1YJ3U 58395383 Ki = 12 nM T86437 CGV59X 58395401 Ki = 0.6 nM T86437 C8KQE6 58395411 Ki = 18 nM T86437 CWR1A7 58395421 Ki = 3.7 nM T86437 C28ADB 58395446 Ki = 0.9 nM T86437 CZR91G 58395466 Ki = 2.1 nM T86437 CLA5V3 58395468 Ki = 21 nM T86437 C0X5CV 58395476 Ki = 2.1 nM T86437 CR9T7W 58438557 IC50 = 44.7 nM T86437 CY3W6B 58438580 IC50 = 272 nM T86437 CR7C4V 58438607 IC50 = 7.4 nM T86437 C9MIL7 58450666 IC50 = 219 nM T86437 CWX4G9 58522116 IC50 = 5090 nM T86437 C4A6LT 58522124 IC50 = 4390 nM T86437 CI9VB0 58522237 IC50 = 3320 nM T86437 C1LE9A 58522238 IC50 = 3470 nM T86437 C74ACR 58522276 IC50 = 8220 nM T86437 CI0L1J 58522322 IC50 = 4160 nM T86437 CVMO97 58522377 IC50 = 3190 nM T86437 C7S1PR 58522381 IC50 = 2150 nM T86437 C8X6YE 58557497 IC50 = 40 nM T86437 C2GO4H 59186418 IC50 = 3055 nM T86437 CPWM60 59291925 IC50 = 22 nM T86437 CE6KO4 59291951 IC50 = 27 nM T86437 CT3EW2 59292007 IC50 = 4.1 nM T86437 C2PE0T 59292008 IC50 = 35 nM T86437 CU3W2S 59292043 IC50 = 50 nM T86437 CC6J4I 59363349 IC50 = 35 nM T86437 CQ93TM 59363383 IC50 = 15 nM T86437 CKQ31B 59363409 IC50 = 42 nM T86437 CW76YC 59589542 IC50 = 1979 nM T86437 C0DV7R 59589757 IC50 = 156 nM T86437 CM50TL 59589801 IC50 > 10000 nM T86437 CZ0LA4 59589877 IC50 = 418 nM T86437 CXJ63M 59603829 IC50 = 4200 nM T86437 CQEU96 59603842 IC50 = 220 nM T86437 C8UMJ2 59617909 Ki > 3500 nM T86437 CDMO01 59617921 Ki > 3500 nM T86437 CUNY05 59617942 Ki = 1700 nM T86437 CY7V3I 59617971 Ki > 3500 nM T86437 CM6B3E 59618010 Ki > 3500 nM T86437 CQCG48 59618036 Ki > 3500 nM T86437 CJ5GF1 59618081 Ki > 3500 nM T86437 CT12JO 59618117 Ki > 3500 nM T86437 C42OZL 59618123 Ki = 490 nM T86437 COI26N 59618146 Ki > 3500 nM T86437 CR5GJ4 59618147 Ki > 3500 nM T86437 C9GB1C 59618160 Ki > 3500 nM T86437 CR9F7D 59618164 Ki = 2900 nM T86437 C7XWE2 59618171 Ki = 1500 nM T86437 C2EIA3 59618285 Ki = 1000 nM T86437 C1ZKR9 59618313 Ki > 3500 nM T86437 C26BNV 59618424 Ki > 3500 nM T86437 C3B7CU 59618428 Ki = 1000 nM T86437 CBH83T 59618445 Ki = 100 nM T86437 C3HC4P 59618462 Ki > 3500 nM T86437 CX0FQ2 59618505 Ki = 200 nM T86437 CG8ET4 59618513 Ki = 2400 nM T86437 CR27IT 59618564 Ki > 3500 nM T86437 CNY59P 60165955 Ki = 0.5 nM T86437 CY3QT8 60165956 Ki = 12 nM T86437 C9PH1Z 60166106 Ki = 50 nM T86437 CR9J1T 60166239 Ki = 11 nM T86437 CO1K2C 60166359 Ki = 33 nM T86437 CEL3B4 60166360 Ki = 6.1 nM T86437 C9IHN3 60166488 Ki = 4.5 nM T86437 C75BLR 60166489 Ki = 5.9 nM T86437 C4FL2P 60166490 Ki = 2.7 nM T86437 C97PZW 60166491 Ki = 9.5 nM T86437 CYK50X 60166623 Ki = 3.2 nM T86437 CKT4Y7 60170769 Ki = 1.2 nM T86437 C3YSV5 60170770 Ki = 9.3 nM T86437 C34RVN 60170771 Ki = 1.5 nM T86437 C74FPI 60170772 Ki = 4.5 nM T86437 CTC8E4 60170773 Ki = 6.1 nM T86437 CR80CH 60170858 Ki = 2.6 nM T86437 C3PA9G 60170859 Ki = 7.3 nM T86437 C2AEG3 60170860 Ki = 90 nM T86437 CHJM71 60170861 Ki = 4.8 nM T86437 CBP48G 60170862 Ki = 5.4 nM T86437 C3R0NO 63107904 IC50 = 24100 nM T86437 CSZ6I5 66556035 IC50 = 501.19 nM T86437 C7MD5X 66556536 IC50 = 1995.26 nM T86437 CNDH38 66557868 Ki = 0.2 nM T86437 CJ08ZL 66604045 IC50 = 49 nM T86437 CY0I2V 66604274 IC50 = 141 nM T86437 CD0LJ6 66604359 IC50 = 52 nM T86437 CS8HK2 66604394 IC50 = 18 nM T86437 C7U8GC 66604464 IC50 = 67 nM T86437 CXU94O 66604576 IC50 = 169 nM T86437 CE9T0V 66604664 IC50 = 1899 nM T86437 C7WO4A 66604791 IC50 = 41 nM T86437 CW53KR 66604810 IC50 = 339 nM T86437 CNW05G 66604855 IC50 = 31 nM T86437 C0JS8O 66604914 IC50 = 5.7 nM T86437 CW9LD1 66604921 IC50 = 62 nM T86437 CTMX20 66605009 IC50 = 31 nM T86437 CP0DB1 66605115 IC50 = 77 nM T86437 CB1WC9 66605298 IC50 = 158 nM T86437 CCWU74 66605322 IC50 = 29 nM T86437 C7Q8ZG 66605359 IC50 = 218 nM T86437 C16TEK 66605475 IC50 = 100 nM T86437 C7MOJ6 66605487 IC50 = 195 nM T86437 CDZA70 66605639 IC50 = 432 nM T86437 C53NBQ 66605756 IC50 = 45 nM T86437 C5PVB2 67008690 IC50 = 2076 nM T86437 C8OZ6W 67008828 IC50 = 863 nM T86437 C1HSE0 67035086 IC50 = 260 nM T86437 CWI6K5 67035106 IC50 > 10000 nM T86437 C38RGB 67035556 IC50 > 10000 nM T86437 CV3HW2 67035568 IC50 > 10000 nM T86437 CZX1E0 67123420 IC50 > 10000 nM T86437 C0RCI2 67123577 IC50 = 5.5 nM T86437 CV63UL 67240318 IC50 > 10000 nM T86437 C78TXA 67277273 IC50 = 110 nM T86437 C0O7TC 67277276 IC50 = 1.5 nM T86437 C3YK7Q 67277763 IC50 = 300 nM T86437 CF4AB0 67277979 IC50 = 2900 nM T86437 C5U2IW 67278045 IC50 = 430 nM T86437 CS9K0L 67278047 IC50 = 140 nM T86437 C2FW8H 67278142 IC50 = 90 nM T86437 CQRS42 67278151 IC50 = 230 nM T86437 C5V9DZ 67278165 IC50 = 520 nM T86437 CMJ29W 67278195 IC50 = 1000 nM T86437 CVL35U 67278385 IC50 = 110 nM T86437 CKVB79 67278425 IC50 = 28 nM T86437 C2C1RE 67329237 IC50 = 41 nM T86437 CV80IQ 67330694 IC50 = 29 nM T86437 CKMV48 67345882 Ki = 0.8 nM T86437 C16THB 67351896 Ki = 12 nM T86437 CXU7P1 67352101 Ki = 16 nM T86437 C4D9NB 67352386 Ki = 8.4 nM T86437 CFX84K 67352945 Ki = 5.9 nM T86437 C1FLT6 67354280 Ki = 120 nM T86437 C9WY2P 67383875 Ki = 24 nM T86437 C14RKJ 67479440 IC50 = 307 nM T86437 C5WQC2 67502257 IC50 > 1000 nM T86437 CX6S4E 68254533 IC50 = 1500 nM T86437 CYMN23 68260892 Ki = 5.4 nM T86437 C4U1IR 68291322 IC50 = 21 nM T86437 C2P7DB 68291391 IC50 = 71 nM T86437 CRM3S0 68291627 IC50 = 100 nM T86437 C4LKB3 68291752 IC50 = 9 nM T86437 CQ49HB 68291755 IC50 = 5 nM T86437 CXI4L1 68291797 IC50 = 41 nM T86437 C8T5VB 68291830 IC50 = 19 nM T86437 CPRW18 68291866 IC50 = 214 nM T86437 C6UWI3 68291981 IC50 = 34 nM T86437 CYN89R 68292156 IC50 = 61 nM T86437 C76EZC 68292170 IC50 = 62 nM T86437 CGA0W6 68292183 IC50 = 15 nM T86437 C93LZT 68292196 IC50 = 190 nM T86437 C8I7GC 68293638 IC50 > 10000 nM T86437 CD56XK 68293660 IC50 > 10000 nM T86437 CYI75G 68678653 IC50 > 30000 nM T86437 C5DGR9 69036886 IC50 = 10000 nM T86437 CK8DC3 69046862 IC50 = 24 nM T86437 COX56A 69809432 IC50 = 189 nM T86437 CECG39 69809726 IC50 = 103 nM T86437 C92EAC 69811936 IC50 = 71 nM T86437 C0XO1M 69812740 IC50 = 113 nM T86437 CASQ98 70650259 IC50 = 1700 nM T86437 CQ2F8J 70824464 Ki = 2600 nM T86437 CJQA59 70929300 IC50 = 67 nM T86437 CNR2Y9 71061323 IC50 = 54 nM T86437 C51JTW 71061588 IC50 = 9.4 nM T86437 CF69WT 71061828 IC50 = 25 nM T86437 COU2C5 71061858 IC50 = 39 nM T86437 CW9OE6 71061878 IC50 = 12 nM T86437 CK9LZ3 71061981 IC50 = 180 nM T86437 CU1T4P 71061987 IC50 = 41 nM T86437 CJH94D 71062030 IC50 = 5.5 nM T86437 CUW46K 71062043 IC50 = 49 nM T86437 C05VNE 71062076 IC50 = 31 nM T86437 C4AC9U 71212257 IC50 < 0.2 nM T86437 CHO4J2 71212467 Ki = 5.4 nM T86437 C7Y2LB 71230234 Ki = 2 nM T86437 CV0U3C 71230392 Ki = 3 nM T86437 COR71Z 71285696 IC50 = 17 nM T86437 C3ZL5S 71285760 IC50 = 64 nM T86437 CME92O 71285933 IC50 = 10 nM T86437 C2FL6H 71286084 IC50 = 5.5 nM T86437 C14YOJ 71286184 IC50 = 12 nM T86437 CX23BP 71288497 IC50 = 22 nM T86437 CH1AJ3 71288512 IC50 = 0.8 nM T86437 CA1T5H 71288539 IC50 = 38 nM T86437 CYU2Z4 71288594 IC50 = 61 nM T86437 CBY4K0 71288602 IC50 = 31 nM T86437 CWLC45 71288607 IC50 = 51 nM T86437 CDST08 71288618 IC50 = 73 nM T86437 C45HTF 71288693 IC50 = 1 nM T86437 COC20B 71288707 IC50 = 370 nM T86437 C6JD3S 71288724 IC50 = 4.6 nM T86437 COV78A 71288729 IC50 = 16 nM T86437 C8DY1N 71288732 IC50 = 61 nM T86437 C6XVG4 71452457 Ki = 24 nM T86437 CY2CE5 71454218 Ki = 5.3 nM T86437 CPO7Y1 71454973 Ki = 2.8 nM T86437 CB8DN6 71455970 Ki = 43 nM T86437 C70KIC 71455971 Ki = 28 nM T86437 CQ0G3P 71455972 Ki = 10 nM T86437 C8LBN3 71457772 Ki = 13 nM T86437 C9HC1M 71457773 Ki = 0.3 nM T86437 C26IQP 71459692 Ki = 2.1 nM T86437 C7GUC2 71461373 Ki = 3.8 nM T86437 CQT1P4 71461404 Ki = 5.8 nM T86437 CTX94J 71461405 Ki = 4.2 nM T86437 CON21P 71463137 Ki = 12 nM T86437 CZPQ54 71463138 Ki = 3.3 nM T86437 CCN01X 71547862 IC50 > 10000 nM T86437 CVEO06 71558636 IC50 = 262 nM T86437 C07SFW 71600166 IC50 = 11600 nM T86437 CWJ1G4 71600167 IC50 = 863 nM T86437 CVYS15 71617859 IC50 = 28 nM T86437 C7T5LI 71655637 Ki = 745 nM T86437 CT3M4B 71655638 Ki = 198 nM T86437 CSC81X 71655639 Ki = 21 nM T86437 CGO74N 71655708 Ki > 3763 nM T86437 C3U1ZV 71655709 Ki = 4.7 nM T86437 CE1JQ3 71655774 Ki = 12 nM T86437 CX5OU4 71681533 Ki = 3.5 nM T86437 C29FVT 71681534 Ki = 10 nM T86437 C7WQP2 71681535 Ki = 13 nM T86437 CEQM71 71681536 Ki = 16 nM T86437 CV5FB0 71681691 Ki = 1.8 nM T86437 C6JH7K 71681692 Ki = 7.2 nM T86437 C30RQG 71681693 Ki = 2.6 nM T86437 C7D8YL 71681694 Ki = 3.4 nM T86437 CE02VF 71681695 Ki = 2 nM T86437 C64WZP 71681852 Ki = 43 nM T86437 C5N6SR 71681853 Ki = 31 nM T86437 CK93ML 71681854 Ki = 1.1 nM T86437 C5E4OF 71682024 Ki = 1.2 nM T86437 C5QK6S 71727668 IC50 = 23 nM T86437 C8PSM2 71737832 Ki = 235 nM T86437 CW52BU 71943288 IC50 = 33000 nM T86437 C54XWG 72190869 IC50 > 10000 nM T86437 C1N7LQ 72202249 IC50 = 5.1 nM T86437 C6THF4 72374600 Ki = 430 nM T86437 CHK46S 72375658 Ki = 98 nM T86437 COPS30 72375659 Ki = 710 nM T86437 CB9ZL4 72375660 Ki = 120 nM T86437 C0K5IO 72375661 Ki = 75 nM T86437 C7PG8Z 72375662 Ki = 398 nM T86437 CCZO42 72375759 Ki = 644 nM T86437 CEV9X5 72375760 Ki = 151 nM T86437 COE6R4 72375761 Ki = 893 nM T86437 C1G8RD 72375763 Ki = 720 nM T86437 C8SLE9 72375764 Ki = 610 nM T86437 C74WLS 72375765 Ki = 3500 nM T86437 CP2KL5 72375766 Ki > 5600 nM T86437 CT9D3J 72375844 Ki = 2800 nM T86437 CZN81X 72375845 Ki = 453 nM T86437 CXL52K 72375846 Ki = 1200 nM T86437 CAV52F 72375847 Ki = 408 nM T86437 C3QT2E 72375850 Ki = 65 nM T86437 C0UJ9M 72375852 Ki = 151 nM T86437 CNJ03L 72375990 Ki > 3500 nM T86437 C5R0WV 72375991 Ki > 3500 nM T86437 CVUL48 72375992 Ki = 2000 nM T86437 CO8KW2 72375993 Ki > 3500 nM T86437 CN0I2W 72375994 Ki > 3500 nM T86437 C1XD7U 72375995 Ki > 3500 nM T86437 C8BJ4U 72375996 Ki > 3500 nM T86437 C7XFW2 72375997 Ki > 3500 nM T86437 CJB95D 72375998 Ki > 3500 nM T86437 CS5V9L 72376089 Ki > 3500 nM T86437 C37GPL 72376090 Ki > 3500 nM T86437 C9U3WO 72376091 Ki > 3500 nM T86437 CK7F6U 72700776 Ki = 3 nM T86437 CLOE10 72706962 IC50 = 1620 nM T86437 CXD38C 73346480 Ki = 2 nM T86437 C0G5RD 73347974 Ki = 661 nM T86437 CRAW59 73349195 Ki = 1100 nM T86437 C41ZJV 73349520 Ki = 4.6 nM T86437 CJE73Y 73352545 Ki = 280 nM T86437 CPRD59 73352546 Ki = 13 nM T86437 CXT70E 73354035 Ki = 380 nM T86437 CGI13D 73354036 Ki = 313 nM T86437 CL4SD8 73355260 Ki > 3500 nM T86437 CMR72H 73355566 Ki = 440 nM T86437 CPT46O 73355567 Ki = 3200 nM T86437 C04CXF 73355568 Ki = 65 nM T86437 C3G2BM 73357112 Ki = 18 nM T86437 CO6F2B 73357113 Ki = 7 nM T86437 CS41CX 75108409 IC50 = 131 nM T86437 CO0BQ5 76310565 IC50 = 628 nM T86437 C6ZAB2 76310566 IC50 > 10000 nM T86437 C0F6VU 76310567 IC50 = 300 nM T86437 CDO38G 76310568 IC50 > 10000 nM T86437 CL42BQ 76310569 IC50 > 10000 nM T86437 CWI1Q4 76310570 IC50 = 564 nM T86437 C8OY6Q 76310785 IC50 > 100000 nM T86437 CAL3U7 76310788 IC50 > 100000 nM T86437 C7SXJ1 76314208 IC50 = 1060 nM T86437 CSDI71 76314209 IC50 > 10000 nM T86437 C12YAE 76314414 IC50 > 100000 nM T86437 CXF1I3 76317774 IC50 = 4903 nM T86437 CY79VS 76317775 IC50 > 10000 nM T86437 CNK2I1 76317776 IC50 > 10000 nM T86437 CS02NA 76317777 IC50 = 1784 nM T86437 CAHW32 76317778 IC50 = 4819 nM T86437 C97RBS 76317979 IC50 > 100000 nM T86437 C2SMK1 76321491 IC50 > 10000 nM T86437 C2DSX7 76321492 IC50 = 4097 nM T86437 CXA4O1 76325093 IC50 > 10000 nM T86437 CEZ64F 76325209 IC50 = 22 nM T86437 C1AI0J 76325315 IC50 > 100000 nM T86437 CPQA45 76325323 IC50 > 100000 nM T86437 C8GK0H 76328659 IC50 = 11120 nM T86437 CJN89E 76332335 IC50 > 10000 nM T86437 CW1QK4 76332336 IC50 = 423 nM T86437 C2P1MX 76332338 IC50 = 2174 nM T86437 CB5Y0Z 76332540 IC50 > 100000 nM T86437 CB4KQ7 76335967 IC50 = 8640 nM T86437 C84PFQ 76335968 IC50 = 2058 nM T86437 CW1HQ9 76370451 IC50 = 3.9 nM T86437 CD6Y1F 78320046 IC50 = 40 nM T86437 CW08SU 78320048 IC50 = 9 nM T86437 CWI93D 78323836 IC50 = 22 nM T86437 C5UK9L 78323837 IC50 = 14 nM T86437 CQ3EJ1 78324132 IC50 = 28 nM T86437 C7VOX0 78324136 IC50 = 42 nM T86437 CA2Y8L 78324435 IC50 = 51 nM T86437 C4I7WD 78324744 IC50 = 22 nM T86437 CQ2SU8 78673832 IC50 > 30000 nM T86437 CE0W9R 78673833 IC50 > 30000 nM T86437 CPG3A5 86302574 IC50 > 30000 nM T86437 C96EDF 86660048 IC50 = 1000 nM T86437 CC8I0M 86707711 IC50 = 1.9 nM T86437 CW4Z2F 89470642 IC50 = 0.15 nM T86437 CBRF87 89470690 IC50 = 0.24 nM T86437 C7B8OH 89470730 IC50 = 14 nM T86437 CHUO79 89471082 IC50 = 3 nM T86437 CDQ8C6 89471114 IC50 = 0.13 nM T86437 C4G5LP 89471136 IC50 = 33 nM T86437 CX1DZ3 89471497 IC50 = 0.3 nM T86437 CX1MA3 89471556 IC50 = 1.2 nM T86437 C1HW4B 89735655 IC50 = 4300 nM T86437 CG9C6J 89765129 IC50 = 48 nM T86437 C13GOX 89775209 IC50 = 90 nM T86437 C3N6RU 89775221 IC50 = 30 nM T86437 CG5P9A 90153688 IC50 > 50000 nM T86437 CTV52A 90367281 IC50 = 1.5 nM T86437 CY0UC4 90645194 IC50 > 10000 nM T86437 C7EXH8 91755097 IC50 = 0.7 nM T86437 C37IZB 91755098 IC50 = 1.3 nM T86437 C7UAK5 91809175 IC50 > 2000 nM T86437 C8RG6H 91827514 IC50 = 1900 nM T86437 C0Y8ZK 91933875 IC50 > 1000 nM T86437 C64SIO 92042864 IC50 = 896 nM T86437 C9BL4M 92045136 IC50 = 22 nM T86437 CXU1Z2 101043725 IC50 > 2000 nM T86437 C9G5TC 102515538 Ki = 172 nM T86437 CM2C3W 105539869 IC50 = 130 nM T86437 C3ECY5 117625437 IC50 = 16 nM T86437 CZC84D 117769161 IC50 = 1.2 nM T86437 CE7BZ8 117769174 IC50 = 28 nM T86437 CBJ07Q 117769217 IC50 = 3.6 nM T86437 CXHQ08 117769229 IC50 = 1 nM T86437 CS9WO4 117769234 IC50 = 0.9 nM T86437 C61VXQ 117769241 IC50 = 0.9 nM T86437 C1SA9I 117769244 IC50 = 2.2 nM T86437 C0VY7C 117769271 IC50 = 0.5 nM T86437 C6O9BT 117769272 IC50 = 7.2 nM T86437 CSR9B0 117769289 IC50 = 1.2 nM T86437 C2M9CR 117769307 IC50 = 3.3 nM T86437 C7FWS3 117769309 IC50 = 0.9 nM T86437 CYWV32 117769339 IC50 = 6.6 nM T86437 CZV35K 117769346 IC50 = 1.7 nM T86437 C5V6RG 117769349 IC50 = 4.9 nM T86437 C4O1PX 117769362 IC50 = 1.2 nM T86437 CPV4C8 117769365 IC50 = 0.6 nM T86437 CP3MC5 117769379 IC50 = 1.2 nM T86437 C8V6LG 117769392 IC50 = 2 nM T86437 C2NBZ8 117769396 IC50 = 1.3 nM T86437 COV59Y 117769408 IC50 = 0.7 nM T86437 CXJ3I6 117769409 IC50 = 4 nM T86437 C8LTZ6 117769464 IC50 = 2.4 nM T86437 C4KL1Y 117769470 IC50 = 0.8 nM T86437 CQ46WT 117769476 IC50 = 2.3 nM T86437 CSKO30 117769533 IC50 = 6.6 nM T86437 C6XC3W 117769575 IC50 = 0.4 nM T86437 CS95HO 117769592 IC50 = 0.8 nM T86437 C0PIL5 117769623 IC50 = 1.6 nM T86437 CO3DA2 117769866 IC50 = 6.9 nM T86437 CI46CP 117770056 IC50 = 230 nM T86437 C7NI8L 117770083 IC50 = 100 nM T86437 CJ3QC8 117770200 IC50 = 3100 nM T86437 CSD47C 117770482 IC50 = 15 nM T86437 C8SNB9 117770595 IC50 = 91 nM T86437 CJ1V9A 117770654 IC50 = 65 nM T86437 CS8E6M 117770678 IC50 = 370 nM T86437 CM7X9N 117770754 IC50 = 79 nM T86437 C4CFG6 117770831 IC50 = 260 nM T86437 C0X1EQ 117809257 IC50 = 26 nM T86437 CDUH09 117809287 IC50 = 0.6 nM T86437 C8HYU9 117926195 IC50 > 10000 nM T86437 CGQK96 118115537 IC50 = 984 nM T86437 C2OX1Q 118115706 IC50 = 274 nM T86437 CWCO47 118115913 IC50 = 2290 nM T86437 C72LYV 118116131 IC50 = 1400 nM T86437 C4JW5D 118116385 IC50 = 1150 nM T86437 CNX7M9 118473558 IC50 > 2000 nM T86437 CK6Z8O 118475621 IC50 = 49 nM T86437 CIVS69 118475644 IC50 = 11 nM T86437 C17FYA 118475649 IC50 = 495 nM T86437 CE49ZI 118475652 IC50 = 35 nM T86437 C65NIK 118475658 IC50 = 656 nM T86437 C0A9RJ 118475705 IC50 = 24.4 nM T86437 CWQ36P 118475893 IC50 = 731 nM T86437 CN04RH 118475894 IC50 > 3000 nM T86437 C2P0CG 118475938 IC50 = 743 nM T86437 CJYV54 118494221 IC50 > 1000 nM T86437 CLTV08 118690376 IC50 = 16 nM T86437 CRK6J2 118690573 IC50 = 67 nM T86437 CTR74C 118690690 IC50 = 24 nM T86437 CY7BI2 118706214 IC50 > 10000 nM T86437 C2C0AG 118707521 IC50 > 100000 nM T86437 C2DJA0 118707522 IC50 > 100000 nM T86437 CBF28W 118707523 IC50 > 100000 nM T86437 CQ6ON4 118707525 IC50 > 100000 nM T86437 C38UWP 118707526 IC50 > 100000 nM T86437 C64ZQX 118707543 IC50 > 100000 nM T86437 CX58DI 118716791 IC50 > 30000 nM T86437 CD9X2B 118716796 IC50 > 30000 nM T86437 C2YJ0O 118716797 IC50 > 30000 nM T86437 CL3UO9 118716798 IC50 > 30000 nM T86437 C71BAM 118716799 IC50 > 30000 nM T86437 CU4EL6 118716806 IC50 > 30000 nM T86437 CP0IO9 118722564 IC50 = 2225 nM T86437 C5K2QD 118723914 IC50 = 48 nM T86437 C59YJC 118723915 IC50 = 24 nM T86437 C2ON7Y 118723916 IC50 = 270 nM T86437 C5U8WG 118723917 IC50 = 56 nM T86437 C0ZMR8 118723918 IC50 = 67 nM T86437 C4Z5LJ 118723919 IC50 = 150 nM T86437 C85ELI 118723920 IC50 = 50 nM T86437 CGW49X 118723921 IC50 = 110 nM T86437 CXC8K9 118723922 IC50 = 270 nM T86437 CR5JD8 118723923 IC50 = 84 nM T86437 C9W1BU 118723924 IC50 = 250 nM T86437 C2K0MN 118724183 IC50 > 10000 nM T86437 C0G8DY 118724184 IC50 > 10000 nM T86437 CYN2Q5 118724185 IC50 > 10000 nM T86437 C5LR9P 118724186 IC50 = 5740 nM T86437 CXUE02 118724187 IC50 > 10000 nM T86437 C2IYQ8 118724188 IC50 = 413 nM T86437 CQEM50 118724189 IC50 > 10000 nM T86437 C38URV 118724190 IC50 = 371 nM T86437 CDI46A 118724191 IC50 = 2554 nM T86437 C9MG2U 118724192 IC50 = 572 nM T86437 CDH50E 118724193 IC50 > 10000 nM T86437 C7AE5B 118724194 IC50 = 3012 nM T86437 CS61RK 118724197 IC50 = 3098 nM T86437 C6LTE8 118724198 IC50 = 0.6 nM T86437 CP1HW5 118724199 IC50 = 8.3 nM T86437 CR8P2W 118724200 IC50 = 147 nM T86437 CW2G9E 118724201 IC50 = 16 nM T86437 C8JGN7 118868847 IC50 = 19 nM T86437 C3DK1Q 118868914 IC50 = 10 nM T86437 CQ1TL7 118879520 IC50 = 90 nM T86437 CAZO34 118911466 IC50 = 470 nM T86437 C6VAE4 118911477 IC50 = 9 nM T86437 CRQV39 118911480 IC50 = 20 nM T86437 C5Z0XH 118911481 IC50 = 8.5 nM T86437 CG0T1W 118911482 IC50 = 170 nM T86437 COD91F 118911483 IC50 = 230 nM T86437 C5LYI2 118911484 IC50 = 160 nM T86437 CA9P3K 118911491 IC50 = 31 nM T86437 CB81YO 118911492 IC50 = 12 nM T86437 C2DG5M 118911497 IC50 = 1400 nM T86437 CI2EU5 118911501 IC50 = 100 nM T86437 CA3EF6 118911506 IC50 = 20 nM T86437 C9BE2G 118911507 IC50 = 520 nM T86437 C75DOY 118911508 IC50 = 16 nM T86437 CZ3D0U 118911512 IC50 = 420 nM T86437 C1AE4J 118911514 IC50 = 40 nM T86437 CN53SL 118911517 IC50 = 21 nM T86437 CCX4J8 118911542 IC50 = 74 nM T86437 C7R0NJ 118911545 IC50 = 120 nM T86437 CIS3Z5 118911549 IC50 = 1.4 nM T86437 C49PME 118911551 IC50 = 1500 nM T86437 CJT3P9 118911552 IC50 = 120 nM T86437 CX01BU 118911553 IC50 = 170 nM T86437 C0TU7V 118911556 IC50 = 26 nM T86437 C0TX7B 118911557 IC50 = 23 nM T86437 CYI3O6 118911558 IC50 = 15 nM T86437 C28MLV 118911560 IC50 = 53 nM T86437 C49UGI 118911561 IC50 = 34 nM T86437 C9LD1H 118911562 IC50 = 190 nM T86437 CTR8D0 118911563 IC50 = 77 nM T86437 CY5EN8 118911565 IC50 = 6.3 nM T86437 C84BPW 118911566 IC50 = 6.9 nM T86437 CT4MJ8 118911570 IC50 = 5.8 nM T86437 C2AZP5 118911571 IC50 = 9.8 nM T86437 CQ59WD 118911572 IC50 = 29 nM T86437 C2S7MO 118911575 IC50 = 9.4 nM T86437 C45HFX 118911579 IC50 = 500 nM T86437 CCSH64 118911580 IC50 = 150 nM T86437 CB48OQ 118911581 IC50 = 12 nM T86437 CZY2V6 118911582 IC50 = 670 nM T86437 C2PA8M 118911583 IC50 = 13 nM T86437 C70XKA 118911584 IC50 = 180 nM T86437 CD9C1A 118911585 IC50 = 75 nM T86437 CRZ20W 118911587 IC50 = 7.2 nM T86437 CTQ4J9 118911588 IC50 = 9.3 nM T86437 C3QKH8 118911601 IC50 = 17 nM T86437 COY26N 118911635 IC50 = 140 nM T86437 CL3C9A 118911638 IC50 = 69 nM T86437 CN4O2C 118911639 IC50 = 50 nM T86437 C9O4WL 118911640 IC50 = 54 nM T86437 C3SE0K 118911642 IC50 = 85 nM T86437 C5LHC4 118911643 IC50 = 2.8 nM T86437 CPK30A 118911645 IC50 = 790 nM T86437 CYTV80 121284861 IC50 > 2000 nM T86437 CY9M5S 122182022 IC50 = 29 nM T86437 C2MCH6 122182157 IC50 = 84 nM T86437 CK4A6L 122182159 IC50 = 11 nM T86437 CFU15S 122191618 IC50 = 65 nM T86437 CE4F3A 122191619 IC50 = 1700 nM T86437 CAC5U1 122191620 IC50 = 220 nM T86437 CRF2K0 122191625 IC50 = 540 nM T86437 CPY1K9 122191778 IC50 = 2728 nM T86437 C1H4IX 122192065 IC50 = 6100 nM T86437 C98EJO 122192066 IC50 = 11300 nM T86437 CM1XD7 122192067 IC50 = 100 nM T86437 C0MLH5 122192068 IC50 = 2200 nM T86437 CC4T6A 122192069 IC50 = 5700 nM T86437 CGO6M7 122192070 IC50 = 4300 nM T86437 CBP34K 122192071 IC50 = 11600 nM T86437 CA2TF6 122192072 IC50 = 18200 nM T86437 CFY30Z 122192073 IC50 = 2900 nM T86437 CJ09XF 122192074 IC50 = 3700 nM T86437 C6LS8X 122192075 IC50 = 3100 nM T86437 C7DJA5 122192076 IC50 = 9300 nM T86437 CAS86F 122192079 IC50 = 32400 nM T86437 CG7TP0 122192080 IC50 = 8100 nM T86437 C5K8UM 122192081 IC50 = 3400 nM T86437 CS4XB9 122199230 IC50 = 90 nM T86437 CNA45R 122362931 IC50 = 19 nM T86437 CW9BU8 126643886 IC50 = 29 nM T86437 C4BJ8G 126645320 IC50 = 10 nM T86437 CL60VJ 126647240 IC50 = 270 nM T86437 C1XS8H 126647348 IC50 = 3.6 nM T86437 CSJ1G7 126647349 IC50 = 650 nM T86437 C9QCD3 126715362 IC50 < 4 nM T86437 CNPB25 126715363 IC50 = 7600 nM T86437 CY7US6 126715366 IC50 = 120 nM T86437 CJS53A 126715367 IC50 < 6 nM T86437 CX37RN 126715380 IC50 = 70 nM T86437 C2DQU9 126715387 IC50 = 643 nM T86437 CH6YP0 126715392 IC50 = 130 nM T86437 C1QB5R 126715400 IC50 = 7 nM T86437 CG7YQ2 126715454 IC50 < 3 nM T86437 CO2X6J 126715460 IC50 = 8 nM T86437 CR9C1G 127030133 IC50 = 22 nM T86437 CU4AJ8 127037981 IC50 = 317 nM T86437 CA0O1B 127037982 IC50 = 274 nM T86437 C50NKB 127037983 IC50 = 12200 nM T86437 CF8KQ6 127038326 IC50 = 832 nM T86437 C5WV8P 127038327 IC50 = 356 nM T86437 CI8ZB6 127038328 IC50 = 4910 nM T86437 C98DQZ 127038947 IC50 = 173 nM T86437 CQ4OE5 127039917 IC50 = 801 nM T86437 CC1XP0 127040339 IC50 = 199 nM T86437 C8H7JN 127040340 IC50 = 177 nM T86437 CRQS46 127040341 IC50 > 30000 nM T86437 C3B0AP 127040342 IC50 = 4510 nM T86437 C7KLD9 127040660 IC50 = 977 nM T86437 C4JF8H 127040661 IC50 = 4.9 nM T86437 CC9J7R 127040662 IC50 = 34 nM T86437 CP1RY4 127040993 IC50 = 9 nM T86437 C7P5MY 127040994 IC50 = 49 nM T86437 CB23SC 127041238 IC50 = 561 nM T86437 CJ7QW5 127041248 IC50 = 73 nM T86437 C1N6BC 127041249 IC50 = 36 nM T86437 C5SLH0 127041250 IC50 = 275 nM T86437 C28YFA 127041251 IC50 > 30000 nM T86437 CIP84Z 127041549 IC50 = 5230 nM T86437 CQP76E 127041550 IC50 = 2100 nM T86437 C3A1VL 127041551 IC50 > 30000 nM T86437 CEJ97D 127041858 IC50 = 17 nM T86437 C35OPG 127041859 IC50 = 177 nM T86437 CEN15W 127041860 IC50 = 138 nM T86437 C4UBE5 127041861 IC50 = 872 nM T86437 C7Q5YC 127045965 IC50 = 670 nM T86437 CB2SE8 127049004 IC50 = 5300 nM T86437 CS6ZO5 127049005 IC50 = 5400 nM T86437 C1PE9L 127050562 IC50 = 80 nM T86437 CZ5D8C 127050563 IC50 = 7000 nM T86437 CX46RS 127050564 IC50 = 2000 nM T86437 C3LI1J 127050565 IC50 = 150 nM T86437 CG91WC 127052080 IC50 = 90 nM T86437 C0FM1R 130196825 IC50 = 787 nM T86437 CZ13WL 130339268 IC50 = 383 nM T86437 CD4NY1 131839645 IC50 = 0.1 nM T86437 CUO0C5 132156633 IC50 > 10000 nM T86437 CK4FI7 132277003 IC50 = 966 nM T86437 C5CZA1 132578411 IC50 = 444 nM T86437 C75NKQ 134537028 IC50 = 26 nM T86437 CPDT50 134537033 IC50 = 110 nM T86437 C8CKE5 134537037 IC50 = 510 nM T86437 C7H8QW 134537039 IC50 = 19 nM T86437 C0ZY5J 134537043 IC50 = 25 nM T86437 CJDM08 134537050 IC50 = 66 nM T86437 CQ7G4C 134537056 IC50 = 4.1 nM T86437 CQ1NX6 134537061 IC50 = 740 nM T86437 C43CFZ 134537067 IC50 = 170 nM T86437 CELH87 134537071 IC50 = 34 nM T86437 C8DAO7 134537074 IC50 = 1.9 nM T86437 CQ9OU1 134537081 IC50 = 140 nM T86437 CH78PN 134537085 IC50 = 160 nM T86437 CN5P0G 134537092 IC50 = 260 nM T86437 CHY1S4 134537094 IC50 = 110 nM T86437 C8L7UN 134537111 IC50 = 11 nM T86437 C42TFN 134537113 IC50 = 13 nM T86437 C58HUF 134537114 IC50 = 53 nM T86437 C3LRB2 134537119 IC50 = 22 nM T86437 CWU3Z2 134537141 IC50 = 52 nM T86437 CEOW01 134537147 IC50 = 17 nM T86437 C0T7VN 134537152 IC50 = 79 nM T86437 CZD72H 134537156 IC50 = 11 nM T86437 C3HC0S 134537158 IC50 = 11 nM T86437 CTP15L 134537160 IC50 = 70 nM T86437 C6Z9QY 134537161 IC50 = 28 nM T86437 C9ME6L 134537163 IC50 = 14 nM T86437 CEQ15Z 134537167 IC50 = 70 nM T86437 C8N6ZF 134537169 IC50 = 9.5 nM T86437 CXA39D 134537177 IC50 = 19 nM T86437 C97OTS 134537185 IC50 = 62 nM T86437 CHK0V4 134611545 IC50 = 0.14 nM T86437 C20FAE 134611548 IC50 = 0.37 nM T86437 C51PKU 134611580 IC50 = 0.22 nM T86437 CN75GU 134611727 IC50 = 12 nM T86437 C80PJI 134611728 IC50 = 16 nM T86437 C2AN7T 134611886 IC50 > 100000 nM T86437 CFM46L 134812674 IC50 = 358 nM T86437 C2VC5Y 134817793 IC50 < 3 nM T86437 CVF86X 135125189 IC50 = 0.07 nM T86437 C9MCQ0 135138184 IC50 = 0.4 nM T86437 C7V2MJ 135142423 IC50 = 0.54 nM T86437 CLET52 135142442 IC50 = 0.3 nM T86437 CU13RW 135142625 IC50 = 1.2 nM T86437 CM7N0J 135142656 IC50 = 0.92 nM T86437 CG6JI9 135142885 IC50 = 0.25 nM T86437 CQD32R 135143120 IC50 = 0.49 nM T86437 C7PJ6X 135566704 IC50 > 30000 nM T86437 CPHG43 135567142 IC50 = 0.1 nM T86437 C2NRS8 135567293 IC50 = 0.4 nM T86437 C4R1FH 135567294 IC50 = 1.7 nM T86437 CA0R9G 135567295 IC50 = 60 nM T86437 CRI5F3 135839295 IC50 = 6.1 nM T86437 CH8W7B 135839328 IC50 = 68.6 nM T86437 CD32NI 135894059 IC50 = 1351 nM T86437 CJID74 136013449 EC50 = 350 nM T86437 CHA4N2 136013680 IC50 > 10 nM T86437 C1DNM8 136048702 IC50 = 0.7 nM T86437 CL53YD 136048703 IC50 = 0.5 nM T86437 C8PFY0 136048704 IC50 = 0.3 nM T86437 CKC87M 136048705 IC50 = 3.2 nM T86437 C8TA5Y 136048706 IC50 = 26 nM T86437 CM2A3P 136048707 IC50 = 1.6 nM T86437 C76OBL 136048708 IC50 = 5 nM T86437 C75UYC 136048709 IC50 = 5 nM T86437 CA10UT 136048710 IC50 = 10 nM T86437 C1YUD0 136219394 IC50 > 10 nM T86437 CIU8W3 136254389 IC50 > 10 nM T86437 C1P6ZW 136263939 IC50 < 0.1 nM T86437 C0R2IL 136901416 IC50 = 4.365 nM T86437 C5JIR2 136987005 IC50 > 100000 nM T86437 CIJ71W 137028350 IC50 = 100 nM T86437 CS15TL 137028351 IC50 = 3100 nM T86437 CH3M4B 137083628 IC50 > 30000 nM T86437 CJA07O 137083629 IC50 > 30000 nM T86437 C9F8PX 137083630 IC50 > 30000 nM T86437 CE9V4U 137174991 IC50 = 2 nM T86437 C2FLS4 137175037 IC50 = 2 nM T86437 C6V7OD 137175063 IC50 = 0.8 nM T86437 C2KF1R 137175070 IC50 = 3 nM T86437 C5XJ4Q 137175071 IC50 = 6 nM T86437 CA3E0R 137175072 IC50 = 13 nM T86437 C4WET8 137175109 IC50 = 0.4 nM T86437 CM64UH 137175110 IC50 = 0.8 nM T86437 CQX1H3 137175111 IC50 = 1.3 nM T86437 C0YBL9 137175112 IC50 = 7 nM T86437 CP7RH5 137175113 IC50 = 8 nM T86437 CJ94DH 137175128 IC50 = 0.9 nM T86437 C70DIP 137223928 IC50 = 1.8 nM T86437 C9F3KV 137321155 IC50 = 3.37 nM T86437 CJK67W 137321156 IC50 = 125.1 nM T86437 C3Z4AT 137321159 IC50 = 2703 nM T86437 CMY0V2 137321160 IC50 = 422 nM T86437 CWM9S4 137349398 IC50 = 5 nM T86437 CAM8K0 137632226 IC50 = 85 nM T86437 CH9WK1 137632228 IC50 = 1100 nM T86437 C7R2HI 137632648 IC50 = 11 nM T86437 C2I3PY 137633211 IC50 = 264 nM T86437 CJN68H 137633647 IC50 = 10 nM T86437 CF6RH5 137633780 IC50 = 0.04 nM T86437 COE76K 137634328 IC50 = 2.1 nM T86437 C6IU0M 137634461 IC50 = 0.9 nM T86437 CE4DH3 137635161 IC50 = 31 nM T86437 C6JVG9 137635398 IC50 = 17 nM T86437 CMV38W 137635509 IC50 = 1422 nM T86437 CM73AT 137635759 IC50 = 17 nM T86437 CH5SI7 137636771 IC50 = 19 nM T86437 C8I2NQ 137637573 IC50 = 196 nM T86437 C3RF7B 137638414 IC50 = 141 nM T86437 CE0ZF8 137638897 IC50 = 1.3 nM T86437 C50WHR 137641404 IC50 = 39 nM T86437 C2VWE5 137642024 IC50 = 37 nM T86437 CJ6PU9 137642141 IC50 = 2.3 nM T86437 C0RX1Z 137642404 IC50 = 0.4 nM T86437 C9GDQ6 137642740 IC50 = 0.19 nM T86437 C94ELU 137643208 IC50 > 2000 nM T86437 CO83EQ 137643608 IC50 = 26.8 nM T86437 CQP79B 137643915 IC50 = 12 nM T86437 CGHP09 137645020 IC50 = 0.9 nM T86437 CN34SE 137646319 IC50 > 2000 nM T86437 CI8S5A 137646690 IC50 = 144 nM T86437 CGE91V 137646834 IC50 = 36 nM T86437 CE8SH2 137647292 IC50 = 974 nM T86437 CW6D9H 137648009 IC50 = 92 nM T86437 C9KW2L 137648948 IC50 = 123 nM T86437 CHN7A3 137648975 IC50 = 8 nM T86437 CIB60Q 137649981 IC50 = 0.24 nM T86437 CF4X3E 137650150 IC50 = 2756.5 nM T86437 CVHT54 137650515 IC50 = 14 nM T86437 CJQ72A 137650866 IC50 = 863 nM T86437 CA9K6R 137650880 IC50 = 52 nM T86437 COCF21 137651256 IC50 = 6 nM T86437 C3Z7LM 137651481 IC50 = 0.5 nM T86437 CQ27PY 137651710 IC50 = 7.5 nM T86437 CYA52Z 137652173 IC50 = 24 nM T86437 C28QUP 137652864 IC50 > 10000 nM T86437 C6UEB9 137653042 IC50 = 30 nM T86437 CK81UT 137654424 IC50 = 1700 nM T86437 CW6SO7 137654686 IC50 = 178 nM T86437 CCR5B3 137654793 IC50 = 11 nM T86437 CKM89A 137654900 IC50 = 0.18 nM T86437 C26ONG 137654955 IC50 = 5 nM T86437 CP5S6L 137655441 IC50 = 0.6 nM T86437 CVBS03 137656215 IC50 = 0.06 nM T86437 CYWE21 137656346 IC50 = 0.5 nM T86437 C6V3WR 137656619 IC50 = 3 nM T86437 CT1EP3 137656679 IC50 = 9.7 nM T86437 C8VC9A 137657080 IC50 = 0.8 nM T86437 C49GYQ 137658008 IC50 = 21 nM T86437 C59BVH 137658028 IC50 = 0.3 nM T86437 CO6C8I 137658504 IC50 = 11 nM T86437 CW4CK8 137659037 IC50 = 1.4 nM T86437 C86KOS 137659382 IC50 = 6 nM T86437 CR41KW 137660124 IC50 = 0.1 nM T86437 CQ8KF2 137660642 IC50 = 70 nM T86437 COMQ54 137661391 IC50 = 15 nM T86437 CJ52WM 137661888 IC50 = 57 nM T86437 CU2L5H 138108525 IC50 = 52 nM T86437 C2W0JU 138319690 EC50 = 30 nM T86437 C28PJZ 138376574 IC50 = 180 nM T86437 CXV84M 138377596 IC50 = 4.8 nM T86437 C8X9DR 138584993 IC50 = 30.17 nM T86437 C9NL1M 138585023 IC50 = 6.59 nM T86437 CHX6N7 138585027 IC50 = 1.2 nM T86437 C3RM2Z 138585033 IC50 = 4.23 nM T86437 CBF8S4 138585069 IC50 = 616.3 nM T86437 C4O0GC 138585070 IC50 = 9.89 nM T86437 C7KYU3 138585074 IC50 = 43.78 nM T86437 CE5S4Z 138585101 IC50 = 3334 nM T86437 CM63FA 138585111 IC50 = 11.48 nM T86437 C2U8PZ 138585129 IC50 = 1.91 nM T86437 C0Y2WZ 138585150 IC50 = 95.62 nM T86437 CHMX08 138585151 IC50 = 17.86 nM T86437 CA8N5T 138585156 IC50 = 37.54 nM T86437 CG8TR3 138585164 IC50 = 5.28 nM T86437 C3JR7K 138585184 IC50 = 138.1 nM T86437 CQI78V 138585192 IC50 = 10.61 nM T86437 C2UCN9 138605457 IC50 = 103.15 nM T86437 C3RM1U 138605458 IC50 = 423.8 nM T86437 CD4M3W 138605461 IC50 = 58.26 nM T86437 C4VMQ9 138605557 IC50 = 304.45 nM T86437 CQ6R7X 138911330 IC50 > 40000 nM T86437 CI1D9F 139600335 IC50 = 26 nM T86437 CI7C4P 140943115 IC50 > 2000 nM T86437 C7U3KH 140943149 IC50 > 2000 nM T86437 C18QDP 141523774 IC50 = 589.1 nM T86437 CD9F4Y 141523776 IC50 = 168.3 nM T86437 C4L6JD 141523781 IC50 = 361.2 nM T86437 CSZQ36 141523784 IC50 = 140 nM T86437 CTYQ49 141523785 IC50 = 190.4 nM T86437 CU51PI 141531440 IC50 = 694 nM T86437 C81RPA 141531442 IC50 = 1946.9 nM T86437 CAT46B 141531443 IC50 = 618.1 nM T86437 CS37YV 141531444 IC50 = 1372.5 nM T86437 CN75MA 141728817 IC50 = 10 nM T86437 C7EL5X 141728840 IC50 = 14 nM T86437 C9H8PX 141728841 IC50 = 15 nM T86437 CC03XH 141728860 IC50 = 30 nM T86437 CECS13 141753441 IC50 = 1286 nM T86437 C1JR5B 142379949 IC50 = 0.14 nM T86437 C45HDA 142744326 IC50 = 82 nM T86437 CFY17M 142744351 IC50 = 138 nM T86437 CM0BL5 142744356 IC50 = 186 nM T86437 C47YDW 142744361 IC50 = 72 nM T86437 C2L1ZB 142744367 IC50 = 142 nM T86437 CZ6FC4 145362469 IC50 = 16 nM T86437 C2OA9H 145949725 IC50 < 3 nM T86437 CY04PB 145950223 EC50 = 37 nM T86437 CDTW63 145950378 IC50 < 3 nM T86437 CDJ81U 145952312 EC50 = 325 nM T86437 C2XP8N 145953005 IC50 = 29 nM T86437 CN0V3D 145953512 EC50 = 68 nM T86437 C1OQ3J 145953599 IC50 < 3 nM T86437 CNS52L 145954024 EC50 = 189 nM T86437 CRU9F8 145955362 IC50 <= 3 nM T86437 CIP2J9 145955397 IC50 = 55 nM T86437 CQ68WS 145956107 IC50 = 4 nM T86437 CZ0B7A 145956262 IC50 = 13 nM T86437 CO6SV3 145957001 IC50 = 42 nM T86437 C51ADW 145958260 IC50 = 10 nM T86437 C3L8IE 145958641 IC50 = 69 nM T86437 C7B2LD 145959014 IC50 < 3 nM T86437 CO05IK 145959360 IC50 = 76 nM T86437 CMCG17 145959462 IC50 < 3 nM T86437 C2LD5V 145960573 EC50 = 101 nM T86437 CFY21D 145961655 EC50 = 7660 nM T86437 CI9Z7U 145962747 IC50 = 45 nM T86437 CQ86LZ 145963345 IC50 = 117 nM T86437 CEDZ18 145971190 EC50 = 26 nM T86437 CKPM09 145971514 IC50 = 6 nM T86437 C7K1AJ 145971681 IC50 = 359 nM T86437 C7OD0E 145973587 EC50 = 50 nM T86437 CHVD06 145979212 IC50 > 10000 nM T86437 C7L1IC 145979240 IC50 = 4027 nM T86437 CAJ37B 145979552 IC50 = 94 nM T86437 CE31VG 145979714 IC50 = 82 nM T86437 C7N8DU 145980127 IC50 = 814 nM T86437 C8AMK1 145980722 IC50 = 100 nM T86437 C81XFH 145980840 IC50 = 105 nM T86437 C85XBC 145981348 IC50 = 81 nM T86437 C5VF8P 145983087 IC50 = 1067 nM T86437 CS1GK8 145983460 IC50 = 146.8 nM T86437 CG97VS 145983548 IC50 = 496.8 nM T86437 CA20KM 145983867 IC50 = 1354.7 nM T86437 C7THN1 145984160 IC50 = 844 nM T86437 C30EHD 145984172 IC50 = 1720 nM T86437 CP8J3H 145984569 IC50 = 112.3 nM T86437 C42SJR 145984669 IC50 = 496.8 nM T86437 CLH7K9 145984673 IC50 = 165.4 nM T86437 C67HUC 145984822 IC50 = 342.4 nM T86437 CG4U3I 145985120 IC50 = 1674.7 nM T86437 CY7X5L 145986106 IC50 = 2291.5 nM T86437 C03PYD 145986466 IC50 < 1000 nM T86437 C2JCA0 145987101 IC50 = 203 nM T86437 CW7V1O 145987719 IC50 > 50000 nM T86437 C8NEY2 145987871 IC50 = 97 nM T86437 C9ZC0H 145987988 IC50 > 2000 nM T86437 C9KJ1A 145988137 IC50 = 94 nM T86437 C9BX4U 145988956 IC50 = 733 nM T86437 CIVK73 145989244 IC50 = 775 nM T86437 CC8GZ3 145989610 IC50 = 113 nM T86437 C5I8SR 145989639 IC50 = 6501 nM T86437 CIU9W4 145990027 IC50 = 369 nM T86437 C3DWZ0 145990496 IC50 > 4163 nM T86437 CTX1A3 145990814 IC50 = 37 nM T86437 CNG35K 145991262 IC50 = 493 nM T86437 C0M6LD 145991292 IC50 = 1715 nM T86437 CKGE38 145991618 IC50 = 1179 nM T86437 CI8R6P 145992803 IC50 = 1942 nM T86437 CD09RT 145992905 IC50 = 52.1 nM T86437 CG21JZ 145993080 IC50 > 2000 nM T86437 CR2F1Y 145993348 IC50 = 92 nM T86437 C51DMH 145993445 IC50 = 652 nM T86437 C1S2ER 146025986 IC50 = 18 nM T86437 CHQU21 146185142 IC50 = 1223 nM T86437 C71KXB 146185156 IC50 = 82 nM T86437 C9IA1X 146185163 IC50 = 1796 nM T86437 CS0OL6 146185170 IC50 = 660 nM T86437 C1IAH7 146185174 IC50 = 120 nM T86437 C5T7UA 154701267 IC50 = 26 nM T86437 C7PLT9 155510967 IC50 = 7179 nM T86437 C1WRE2 155511764 IC50 = 76 nM T86437 CR1SE8 155511850 IC50 = 3062 nM T86437 C2MD1Q 155513187 IC50 > 10000 nM T86437 CM95KR 155513637 IC50 = 627.1 nM T86437 C83ZSG 155514311 IC50 = 30 nM T86437 C7MJY5 155514805 IC50 = 21 nM T86437 CUIO35 155516044 IC50 = 215 nM T86437 CTP29J 155516678 IC50 = 20 nM T86437 C9VK3I 155517004 IC50 > 2000 nM T86437 C2X8HA 155517088 IC50 > 2000 nM T86437 CE2Q3D 155517448 IC50 = 70 nM T86437 C0E7WS 155518120 IC50 = 234 nM T86437 CDTG10 155518349 IC50 = 4 nM T86437 CQ19HO 155518921 IC50 = 4 nM T86437 CLK4S9 155519594 IC50 = 1510 nM T86437 CF0H9V 155520176 IC50 = 124 nM T86437 C0A9LX 155520276 IC50 > 10000 nM T86437 C4YJN9 155520341 IC50 = 17 nM T86437 C1PJC7 155520619 IC50 = 130 nM T86437 C0YEX7 155521332 IC50 = 38 nM T86437 CXG4L3 155522806 IC50 = 3.4 nM T86437 C9LUO3 155523352 IC50 = 43 nM T86437 C7NVQ5 155523535 IC50 = 380.2 nM T86437 C32POG 155523862 IC50 = 996.2 nM T86437 CE4FX7 155525956 IC50 = 469.2 nM T86437 CCS24O 155527492 IC50 = 2630.4 nM T86437 CK14UT 155528172 IC50 = 748 nM T86437 CB26JT 155528364 IC50 = 33 nM T86437 CVW07K 155528897 IC50 = 121 nM T86437 CL47NH 155529550 IC50 = 180 nM T86437 CRX08F 155531665 IC50 = 260 nM T86437 CQU09F 155532106 IC50 = 27 nM T86437 C5V6PY 155532206 IC50 > 2000 nM T86437 C4LE7Q 155532724 IC50 = 23 nM T86437 CLSV71 155533995 IC50 = 110 nM T86437 CGH63O 155534464 IC50 = 1.9 nM T86437 C2NPE6 155534808 IC50 = 110 nM T86437 C64FIW 155534972 IC50 = 842 nM T86437 CE8QW2 155535975 IC50 = 13 nM T86437 CMV7B2 155538485 IC50 = 2400 nM T86437 C5GNH8 155538704 IC50 = 285 nM T86437 C5WB0T 155539358 IC50 = 9670 nM T86437 C03BNT 155539537 IC50 = 10800 nM T86437 C3O6KI 155540160 IC50 = 92 nM T86437 C0D8OL 155540191 IC50 = 28.84 nM T86437 C16MHE 155540242 IC50 > 2000 nM T86437 CBA08W 155540345 IC50 = 11500 nM T86437 CP2NY0 155540484 IC50 = 4.169 nM T86437 CF8O5T 155540488 IC50 = 831.76 nM T86437 C51JNT 155540621 IC50 = 5.495 nM T86437 C76QBR 155541045 IC50 = 2200 nM T86437 CT1AX5 155541077 IC50 = 6.918 nM T86437 CY8F7S 155541097 IC50 = 104 nM T86437 CH6LV1 155541475 IC50 = 70.79 nM T86437 CS58BA 155541478 IC50 = 920 nM T86437 CF9AX3 155542099 IC50 = 750 nM T86437 C1B6EK 155542401 IC50 = 25.12 nM T86437 CH59RW 155542578 IC50 = 13 nM T86437 CKL31P 155542961 IC50 = 69.18 nM T86437 CH46TG 155543289 IC50 = 643 nM T86437 C1QRZ2 155543349 IC50 = 14 nM T86437 CKM8G4 155543489 IC50 = 1821 nM T86437 CRA21U 155543538 IC50 = 1159 nM T86437 CD9Z3W 155544141 IC50 = 8.7 nM T86437 CZ3YI6 155544372 IC50 = 943 nM T86437 CTQ63L 155544706 IC50 = 33.88 nM T86437 CP7XE1 155545114 IC50 = 29.51 nM T86437 CFR42U 155545338 IC50 = 104.71 nM T86437 C5BHW8 155546008 IC50 = 43 nM T86437 C5U8HP 155546232 IC50 = 37.15 nM T86437 CJ8F7V 155546474 IC50 = 33900 nM T86437 CSI1U9 155547916 IC50 = 81 nM T86437 C0B3RK 155547921 IC50 = 169.82 nM T86437 C3DZU0 155548345 IC50 = 40 nM T86437 CPR01A 155549631 IC50 = 2270 nM T86437 CI6Y5Z 155549690 IC50 = 3.981 nM T86437 C10OSG 155550219 IC50 = 40 nM T86437 C3DW8J 155550308 IC50 = 9.333 nM T86437 C31QUW 155550462 IC50 = 32 nM T86437 C6UJS7 155550600 IC50 = 200 nM T86437 C0DMP2 155551420 IC50 = 1240 nM T86437 CHM8G1 155551600 IC50 = 22000 nM T86437 C2Q1LR 155552255 IC50 = 20 nM T86437 CW1UX0 155552333 IC50 = 11.48 nM T86437 CV4NX3 155552736 IC50 = 7940 nM T86437 C62ERW 155552853 IC50 = 31.62 nM T86437 CPB6M8 155553409 IC50 = 923 nM T86437 C5HQ7X 155553551 IC50 = 6 nM T86437 CADO35 155554376 IC50 = 414 nM T86437 CNTP52 155554413 IC50 = 63 nM T86437 CWLC85 155554605 IC50 = 104 nM T86437 CQ6S8E 155554939 IC50 = 16.6 nM T86437 C47MNG 155554972 IC50 = 1100 nM T86437 CP39ZD 155555305 IC50 = 295.12 nM T86437 C9J4HM 155555486 IC50 = 3473 nM T86437 CTRV23 155555922 IC50 = 460 nM T86437 C2VS8X 155556321 IC50 = 1319 nM T86437 CG48UE 155556474 IC50 = 9.12 nM T86437 C8TYG7 155556520 IC50 > 9524 nM T86437 C59HKP 155557055 IC50 > 3000 nM T86437 CH9ON1 155557340 IC50 = 1242 nM T86437 CZUT98 155557375 IC50 = 460 nM T86437 CG9E7Z 155557901 IC50 = 151 nM T86437 CHW4O3 155558352 IC50 = 16.6 nM T86437 C7HFI8 155558403 IC50 = 47 nM T86437 C2LK9V 155558426 IC50 = 2032 nM T86437 C7WND0 155558729 IC50 = 199 nM T86437 C3V5HL 155559143 IC50 = 96.2 nM T86437 C2U5ZM 155559343 IC50 = 34.67 nM T86437 CSF54R 155559609 IC50 = 1262 nM T86437 CANJ25 155559746 IC50 = 851.14 nM T86437 C46KLS 155559780 IC50 > 1000 nM T86437 CNK81M 155560413 IC50 = 54.95 nM T86437 C54NQC 155561203 IC50 = 76 nM T86437 C1Z6IL 155561218 IC50 = 90 nM T86437 CH1LJ2 155562424 IC50 = 1586 nM T86437 CRU0K3 155563465 IC50 = 9290 nM T86437 C68TCL 155563799 IC50 = 774 nM T86437 C1NM2T 155564180 IC50 = 1820 nM T86437 CBQN81 155564466 IC50 = 1126 nM T86437 CZ2NK9 155565077 IC50 = 2884.03 nM T86437 CA0Z1U 155565486 IC50 = 21600 nM T86437 CSNF76 155565806 IC50 = 14.13 nM T86437 CF1X5I 155566525 IC50 = 122 nM T86437 C7S5MC 155566661 IC50 > 3000 nM T86437 CQA46B 155566981 IC50 = 10500 nM T86437 C6AXL1 155567447 IC50 = 2610 nM T86437 CSRZ04 155567801 IC50 > 3000 nM T86437 CGX28M 155567987 IC50 = 1700 nM T86437 COS7X5 155568028 IC50 = 253.8 nM T86437 COGC41 155568181 IC50 = 287.4 nM T86437 C0L6UT 155568261 IC50 = 19.05 nM T86437 CR79DJ 155568314 IC50 > 3000 nM T86437 C8EYW3 155568955 IC50 = 852 nM T86437 CRHE56 155569596 IC50 = 8800 nM T86437 CE50IC 155569626 IC50 = 3300 nM T86437 C3X6WU 155569641 IC50 = 764 nM T86437 C14DIR 16750188 IC50 = 3000 nM T86437 C5UI4F 16750189 IC50 = 5800 nM T86437 C6JKT9 16750206 IC50 > 10000 nM T86437 CYIU14 16750228 IC50 = 3500 nM T86437 CX4I6T 16750253 IC50 = 1700 nM T86437 CI79TY 16750254 IC50 = 8700 nM T86437 CS6UT4 16750288 IC50 = 3600 nM T86437 COM3C1 16750290 IC50 = 4600 nM T86437 CI67WG 16750292 IC50 = 1000 nM T86437 CIGJ63 16750308 IC50 = 3600 nM T86437 CL2SY5 16750330 IC50 = 4900 nM T86437 CE5P2I 53363072 IC50 = 2500 nM T86437 CTV60O 53363073 IC50 = 3100 nM T86437 CD74BW 53363074 IC50 = 2800 nM T86437 CU3M8P 53363075 IC50 > 10000 nM T86437 C07FTA 53363076 IC50 > 10000 nM T86437 C9JX2G 53363150 IC50 = 950 nM T86437 CJ04SF 53363151 IC50 = 1300 nM T86437 CO7Z2P 53363152 IC50 = 940 nM T86437 C1T2LY 53363154 IC50 = 2100 nM T86437 C9GEA7 53363242 IC50 = 2400 nM T86437 CTSP38 53363245 IC50 = 1900 nM T86437 CM7BZ3 53363246 IC50 = 830 nM T86437 C0QON7 53363337 IC50 = 380 nM T86437 CU76JB 53363338 IC50 > 10000 nM T86437 C2PU3M 53364335 IC50 > 10000 nM T86437 C10FXI 53364337 IC50 = 1900 nM T86437 C2U9QE 53364338 IC50 = 400 nM T86437 D02BXJ 46864270 IC50 = 55.3 nM T86437 D03BQI 3794 IC50 > 10000 nM T86437 D06HVH 54613583 IC50 > 10000 nM T86437 D09HVH 135566652 IC50 > 10 nM T86437 D0E5IP 3795 IC50 > 10000 nM T86437 D0H7DQ 6419755 IC50 = 770 nM T86437 D0IR6U 5494425 IC50 = 4 nM T86437 D0US9O 45275255 IC50 < 3 nM T86437 D0V6VQ 53344620 IC50 = 37.5 nM T86437 D0VC0I 5169 IC50 > 100000 nM T86399 D02YNI 9936746 Ki = 5.4 nM T86399 D05ICT 132010322 Ki = 4.6 nM T86399 D07OFM 46943432 IC50 = 32.5 nM T86399 D0M2TS 71600087 Ki = 1 nM T86399 D0PH9I 118693659 Ki = 100 nM T86399 D0ZW4W 46907787 Ki = 12.5 nM T86399 D09SFV 3973 IC50 = 10300 nM T86399 C92EYR 1503595 IC50 = 30000 nM T86399 C8BZ9Y 5325760 IC50 = 34300 nM T86399 CIG94A 13953713 IC50 = 25118.86 nM T86399 CO6HM1 16480179 IC50 = 22000 nM T86399 C3UFS6 39791103 IC50 = 3000 nM T86399 C2P0IW 44243549 IC50 = 6000 nM T86399 C3VRO9 44557921 IC50 > 10000 nM T86399 C98BLM 49871817 IC50 = 16 nM T86399 CG3PR6 52912222 IC50 = 3.162 nM T86399 CBXV52 52932793 IC50 = 199.53 nM T86399 CJE59U 52932930 IC50 = 3162.28 nM T86399 CSZ2T6 52932933 IC50 = 12589.25 nM T86399 CN87IR 52933159 IC50 = 2511.89 nM T86399 CG6OL4 52933160 IC50 = 794.33 nM T86399 CP8Y9K 52933161 IC50 = 1995.26 nM T86399 CK8Z4P 52933165 IC50 = 15848.93 nM T86399 CKC17F 52933403 IC50 = 1584.89 nM T86399 CD08ZX 52933405 IC50 = 3162.28 nM T86399 C1T7VQ 52933407 IC50 = 2511.89 nM T86399 CO8VX9 52933655 IC50 = 3162.28 nM T86399 C6G7BE 52933893 IC50 = 2511.89 nM T86399 C7VN1E 52934039 IC50 = 1584.89 nM T86399 CUZE18 52934122 IC50 = 1995.26 nM T86399 CN16FE 52934128 IC50 = 2511.89 nM T86399 CTS13B 52934275 IC50 = 1584.89 nM T86399 CNOH36 52935183 IC50 = 398.11 nM T86399 CLRH53 52935478 IC50 = 1995.26 nM T86399 CJIB35 53054190 IC50 = 5200 nM T86399 C6V8YR 53054191 IC50 = 14000 nM T86399 C09HTR 53054200 IC50 = 1400 nM T86399 CUS8F7 53054236 IC50 = 4300 nM T86399 CX5QN4 53054237 IC50 = 13000 nM T86399 CD2TY9 53054238 IC50 = 11000 nM T86399 C47GAW 53054240 IC50 = 4900 nM T86399 CVH2G1 53054241 IC50 = 2400 nM T86399 CF9E2V 53054248 IC50 = 2000 nM T86399 CRWK92 53054249 IC50 = 6000 nM T86399 CSXI51 53054250 IC50 = 2500 nM T86399 CM12EL 53054251 IC50 = 2500 nM T86399 CY5L3J 53054252 IC50 = 3600 nM T86399 CWV76Y 53054258 IC50 = 900 nM T86399 CIU8P7 53054259 IC50 = 500 nM T86399 CVX3R0 53054274 IC50 = 3900 nM T86399 CB05OM 53054276 IC50 = 1700 nM T86399 CLR97U 53054289 IC50 = 1500 nM T86399 CJ6E2Q 53054291 IC50 = 4400 nM T86399 C1WSZ4 53054297 IC50 = 2200 nM T86399 C7A2XC 53054319 IC50 = 1800 nM T86399 C0J1EO 53054320 IC50 = 4700 nM T86399 CK68UF 53054321 IC50 = 1100 nM T86399 CJY5S2 53054322 IC50 = 4200 nM T86399 C1YW5L 53054324 IC50 = 1500 nM T86399 C8Q6WG 53054325 IC50 = 1100 nM T86399 CQEF28 53308655 IC50 = 28200 nM T86399 C9V5LX 53318989 IC50 = 160 nM T86399 CEK3X6 54757749 IC50 = 7400 nM T86399 C1D3WH 54757750 IC50 = 4200 nM T86399 C1DZ7Y 54757751 IC50 = 3300 nM T86399 C6W5OZ 54757752 IC50 = 2300 nM T86399 C1KWY4 54759170 IC50 = 2000 nM T86399 C7HK2C 56924692 IC50 = 1500 nM T86399 CX6SD9 56950289 IC50 = 3600 nM T86399 CZ6NE0 56950420 IC50 = 1500 nM T86399 CJ5BE9 56950421 IC50 = 3600 nM T86399 CL96VQ 56950422 IC50 = 1900 nM T86399 CCLD98 56950423 IC50 = 12000 nM T86399 CZD7G2 56950424 IC50 = 5600 nM T86399 CPQ0B7 56950425 IC50 = 8100 nM T86399 CL90DK 56950426 IC50 = 800 nM T86399 CF9IJ1 56950561 IC50 = 800 nM T86399 CH24QC 56950562 IC50 = 14000 nM T86399 CU62NO 56950563 IC50 = 16000 nM T86399 CRD86M 56950564 IC50 = 19000 nM T86399 CNQ2L5 56950565 IC50 = 31000 nM T86399 CB3A1Z 56950566 IC50 = 11000 nM T86399 C5ADP4 56950567 IC50 = 9000 nM T86399 CFW0D1 57339435 IC50 = 794.33 nM T86399 CF8B4E 60498769 IC50 = 59000 nM T86399 CPY59D 67195867 IC50 = 50118.72 nM T86399 CN3KZ8 68161075 IC50 = 501.19 nM T86399 C49IOA 68161669 IC50 = 794.33 nM T86399 CJ7N3M 68184870 IC50 = 1258.93 nM T86399 CT4Z2A 68184871 IC50 = 630.96 nM T86399 CEX74I 68186034 IC50 = 10000 nM T86399 C25INY 68204735 IC50 = 2511.89 nM T86399 CMC7V5 70664240 IC50 = 1995.26 nM T86399 C1I6OH 70681167 IC50 = 12589.25 nM T86399 C7GJW9 70681170 IC50 = 501.19 nM T86399 C8H4JX 70681173 IC50 = 1000 nM T86399 C6NYK2 70681174 IC50 = 501.19 nM T86399 C8KBJ0 70683271 IC50 = 1995.26 nM T86399 CXD3F9 70691699 IC50 = 501.19 nM T86399 CL8Y9N 71450297 IC50 = 1584.89 nM T86399 C6CQT5 71462842 IC50 = 3162.28 nM T86399 CIPN50 71760902 Ki = 14 nM T86399 C2AFW1 72702849 IC50 = 1258.93 nM T86399 C3R1IL 72703043 IC50 = 100000 nM T86399 CK9O6W 72705811 IC50 = 31622.78 nM T86399 C5TB9S 77843982 Ki = 27 nM T86399 CS6XE0 77846025 Ki = 11.1 nM T86399 COZ8S1 78319129 Ki = 160 nM T86399 C4IF8T 78425807 Ki = 0.48 nM T86399 CFE7R3 86270928 Ki = 2.5 nM T86399 C53QEW 86669224 IC50 = 15848.93 nM T86399 CEDL57 89657555 IC50 = 16 nM T86399 CZJ8W9 90387575 Ki = 15.4 nM T86399 CU91GC 105539824 IC50 = 20000 nM T86399 C1W3XP 112499930 IC50 = 1600 nM T86399 CYX7T2 117072549 IC50 > 100000 nM T86399 CPN74M 118719856 IC50 = 794.33 nM T86399 CE8DL3 118719857 IC50 = 1000 nM T86399 COEU47 118719858 IC50 = 1995.26 nM T86399 CX05SW 118719859 IC50 = 1258.93 nM T86399 CRCG07 118719860 IC50 = 794.33 nM T86399 C03XDG 118719861 IC50 = 794.33 nM T86399 C3ML2F 118719862 IC50 = 1258.93 nM T86399 CZ67WF 118719863 IC50 = 25118.86 nM T86399 C0HR9Y 118719864 IC50 = 501.19 nM T86399 C7F4EP 118719865 IC50 = 1000 nM T86399 CA40QV 118719866 IC50 = 1258.93 nM T86399 CZ8QI6 118719867 IC50 = 1584.89 nM T86399 C8NRI9 118719868 IC50 = 1258.93 nM T86399 C3Y2WT 118719869 IC50 = 1584.89 nM T86399 C52HPM 118719870 IC50 = 630.96 nM T86399 CUT97H 118719871 IC50 = 630.96 nM T86399 CBE68N 118719872 IC50 = 1000 nM T86399 C29WRE 118719873 IC50 = 794.33 nM T86399 C8J0TY 118719874 IC50 = 1995.26 nM T86399 CZR10C 118719875 IC50 = 3981.07 nM T86399 C35AWU 118719876 IC50 = 6309.57 nM T86399 C87ZPY 118796358 IC50 > 100000 nM T86399 C9MQF0 119098887 IC50 = 33234 nM T86399 C0QX4D 119098889 IC50 = 50857 nM T86399 C4ITM8 122180892 IC50 = 23000 nM T86399 CFCA87 122180893 IC50 = 24000 nM T86399 CZRJ29 122180894 IC50 = 13000 nM T86399 C8RE2M 122180895 IC50 > 50000 nM T86399 C54NBV 122180896 IC50 = 13000 nM T86399 C26RAL 122180897 IC50 = 26000 nM T86399 CC35RW 122180898 IC50 = 5000 nM T86399 C7E3VM 122180899 IC50 = 25000 nM T86399 C2UQW0 122180900 IC50 > 50000 nM T86399 C67LPS 122180901 IC50 = 10000 nM T86399 C3FC0Z 122180902 IC50 = 12000 nM T86399 CSR48T 122180903 IC50 = 49000 nM T86399 CVI96R 122180904 IC50 > 50000 nM T86399 CXP8T3 122180909 IC50 = 12000 nM T86399 C3QJ5L 122181550 IC50 > 31622.78 nM T86399 CLI1P6 122235215 EC50 = 480 nM T86399 C4GYP3 126521168 IC50 = 43 nM T86399 CL2PG5 126521180 IC50 = 52 nM T86399 CQV90I 126521354 IC50 = 185 nM T86399 C0HJV7 126521430 IC50 > 999 nM T86399 CN6FI1 126521537 IC50 = 6 nM T86399 C1DOG4 126521586 IC50 = 25 nM T86399 CRY0S6 126563516 IC50 = 38 nM T86399 CN0D6M 126563562 IC50 = 34 nM T86399 CKB36S 126563576 IC50 = 25 nM T86399 CX79NH 126563597 IC50 = 44 nM T86399 C2K5XG 126563611 IC50 = 95 nM T86399 CZ06NR 126563612 IC50 = 45 nM T86399 CM5P2Z 126563615 IC50 = 40 nM T86399 C15ILF 126564427 IC50 = 28 nM T86399 CROY39 126564463 IC50 = 25 nM T86399 CHO12Y 126564469 IC50 > 10000 nM T86399 CB2AS4 126564470 IC50 = 33 nM T86399 CBW08I 126564471 IC50 = 39 nM T86399 CD78GB 126564481 IC50 = 25 nM T86399 CU8CA9 126564486 IC50 = 17 nM T86399 CQW6P1 126564822 IC50 = 24 nM T86399 CQS5T2 126564831 IC50 = 204 nM T86399 CNP2L7 126564832 IC50 = 18 nM T86399 C58PNK 126564833 IC50 = 37 nM T86399 CHPV09 126564847 IC50 = 3 nM T86399 CJZW04 126564858 IC50 = 20 nM T86399 CH14FC 127032939 IC50 = 6600 nM T86399 CS4NG8 127033568 IC50 = 30000 nM T86399 CGA71L 127048256 IC50 = 59555 nM T86399 CH6T5J 127048257 IC50 = 30330 nM T86399 C60SZQ 127048258 IC50 = 21687 nM T86399 C50BMV 127049279 IC50 = 5876 nM T86399 CTF4N2 127051087 IC50 > 100000 nM T86399 CLSZ47 127051725 IC50 = 16654 nM T86399 CMY93U 127051726 IC50 > 100000 nM T86399 CY8V1A 127051727 IC50 > 100000 nM T86399 CXZT48 127052023 IC50 > 100000 nM T86399 C9L1OG 130345579 Ki = 1.7 nM T86399 CTDG89 135141500 IC50 = 830 nM T86399 CF2BU6 135141501 IC50 = 410 nM T86399 CBC37Z 135141502 IC50 = 1910 nM T86399 C12HJT 135141503 IC50 = 1400 nM T86399 C50NEZ 135141504 IC50 = 1080 nM T86399 CRNY32 135397673 Ki = 0.27 nM T86399 C5F3LV 135567026 IC50 = 24600 nM T86399 CO71RI 137285009 IC50 = 1836 nM T86399 CS9MR6 137285011 IC50 = 803 nM T86399 CFXE14 137321203 IC50 = 100 nM T86399 CXN4U1 137321204 IC50 = 316.23 nM T86399 C4VNB8 137369426 IC50 = 147 nM T86399 CU5N8O 137701509 IC50 = 29000 nM T86399 CQ6XB7 139030526 IC50 = 19952.62 nM T86399 C1G9LA 139035062 Ki = 3.1 nM T86399 CG6X3A 142535938 IC50 = 35 nM T86399 CD6U7X 145925666 IC50 = 8948 nM T86399 C1HLK5 145951928 IC50 = 44 nM T86399 CV83ED 145972103 Ki = 2.6 nM T86399 CK20BY 145988169 Ki = 57.3 nM T86399 C9FIY4 153534005 IC50 = 16400 nM T86399 CFD6H1 155352361 IC50 = 30000 nM T86399 CFK2B1 155352401 IC50 > 250000 nM T86399 C76QMK 155513141 Ki = 8.9 nM T86399 C27LFN 155514936 IC50 = 1800 nM T86399 C6OP0S 155535292 Ki = 9.1 nM T86399 C0HI7N 155536879 IC50 = 997 nM T86399 CUX25H 155547195 Ki = 19.1 nM T86399 CZA5N1 155561689 IC50 > 45000 nM T86399 C7ICA9 155564455 IC50 = 78 nM T86399 D00XRH 91820725 IC50 = 3981.07 nM T86399 D03LIP 13953710 IC50 = 29.9 nM T86399 D09VHS 3971 IC50 = 7400 nM T86399 D0F5TZ 91827383 IC50 = 6309.57 nM T86399 D0H3TC 54669868 IC50 = 1600 nM T86399 D0T3AT 672548 IC50 = 28000 nM T86399 D0WU1S 52912189 Ki = 9 nM T43332 D00LOB 9866964 Ki > 26000 nM T43332 D01MUU 183797 IC50 = 3300 nM T43332 D03QJN 9895762 Ki > 15000 nM T43332 CZP0Y1 204101 Ki > 15000 nM T43332 CR4KE5 445844 Ki = 1700 nM T43332 CSL82K 449091 Ki = 380 nM T43332 C1C3RE 449247 Ki = 0.35 nM T43332 CPZ6A3 5287506 Ki = 4 nM T43332 CE83KU 5388938 IC50 = 9.4 nM T43332 C7SYK9 6102731 IC50 = 5 nM T43332 C49IOZ 6857707 Ki > 150000 nM T43332 CX34ZD 9549214 Ki > 1800 nM T43332 CH9IE6 9808346 Ki > 100000 nM T43332 C2AXV0 9809479 Ki > 15000 nM T43332 C4KEZ2 9821506 Ki = 160 nM T43332 C2TA1I 9845742 IC50 = 340 nM T43332 CW3EC6 9848592 Ki = 220 nM T43332 CS9HQ0 9850467 IC50 = 200 nM T43332 CZ9LR2 9870910 Ki = 130 nM T43332 C2F5NS 9884570 Ki = 750 nM T43332 C7I5RG 9892392 Ki = 7000 nM T43332 CMC95R 9910164 Ki = 200 nM T43332 CAP0O8 9910540 Ki = 4 nM T43332 CC0D5H 9915041 Ki > 15000 nM T43332 CVND52 9915545 Ki = 12 nM T43332 CC9QH7 9937406 IC50 = 270 nM T43332 C8F5CW 9937921 Ki > 15000 nM T43332 C8LR4T 9938917 Ki > 15000 nM T43332 CX85LD 9954980 Ki > 16000 nM T43332 C3S7IV 9979724 Ki = 93 nM T43332 CK6XE9 9982431 IC50 = 118 nM T43332 CUG6R3 10037159 Ki = 1450 nM T43332 CXZ2V3 10054210 Ki = 4200 nM T43332 CI2KG6 10072299 IC50 = 52 nM T43332 CD0VO9 10078364 IC50 = 42 nM T43332 C8L7HY 10097631 Ki = 86 nM T43332 C31QAL 10143532 Ki > 15000 nM T43332 C4CZ0T 10162659 IC50 = 118 nM T43332 CFIH78 10185526 IC50 = 11 nM T43332 CYR45Q 10227730 IC50 = 500 nM T43332 CL09QG 10349678 IC50 = 200 nM T43332 CL07UC 10364218 Ki = 23 nM T43332 CM6L0W 10389769 Ki = 13 nM T43332 CVK4L6 10418061 IC50 > 100000 nM T43332 C4SZV0 10454685 Ki = 27 nM T43332 CWU81H 10456905 Ki = 50 nM T43332 CEI65Z 10483775 Ki = 629 nM T43332 CBK06L 10861643 IC50 > 100000 nM T43332 C02XLH 10865109 IC50 = 110 nM T43332 C9LEJ0 10865386 IC50 = 2820 nM T43332 C1BOZ5 10865461 IC50 = 230 nM T43332 CN2CE8 10865462 IC50 = 680 nM T43332 CLB15C 10871563 Ki = 7000 nM T43332 C3Z6PT 10874628 IC50 > 30000 nM T43332 C7YEP4 10875960 IC50 = 1450 nM T43332 C2GPU4 10897682 IC50 = 700 nM T43332 CB1HW4 10905809 IC50 = 2500 nM T43332 CPJ1Q7 10908669 IC50 = 170 nM T43332 C9E7RY 10908791 IC50 = 3180 nM T43332 C2BXU9 10908808 IC50 = 570 nM T43332 C5A8NU 10919581 IC50 = 1290 nM T43332 CMK6P8 10928757 IC50 > 30000 nM T43332 C1Q9WZ 10930326 IC50 = 820 nM T43332 CL20KX 10930722 IC50 = 1830 nM T43332 C2TBO9 10959252 Ki = 16000 nM T43332 CCE31H 10963578 IC50 = 170 nM T43332 CH0VN7 10972370 IC50 > 30000 nM T43332 CIU42D 10973463 IC50 > 30000 nM T43332 C6HG4P 10974490 IC50 = 3300 nM T43332 CVT26S 10974535 IC50 = 900 nM T43332 CH41ZW 10974733 IC50 = 9970 nM T43332 CWVR40 10985371 IC50 = 13700 nM T43332 CM5Y6J 10994432 IC50 = 2700 nM T43332 C4VA7K 10994660 IC50 > 30000 nM T43332 CT7L2Q 10996309 IC50 = 800 nM T43332 C8AG4Z 11005226 IC50 > 30000 nM T43332 CFO15P 11015356 IC50 = 16400 nM T43332 CD4LJ1 11027118 IC50 > 30000 nM T43332 C2RG6V 11028969 IC50 = 190 nM T43332 C7RM5W 11039881 IC50 = 160 nM T43332 C7P5EN 11039916 IC50 = 5880 nM T43332 C4UY7P 11050903 IC50 = 1950 nM T43332 CQ61ZR 11059085 IC50 > 30000 nM T43332 C8L9KE 11059896 IC50 = 3980 nM T43332 C7YDH0 11072681 IC50 = 500 nM T43332 C9CUO6 11102065 IC50 = 14700 nM T43332 CU53EA 11104490 IC50 = 200 nM T43332 CANW92 11112933 IC50 > 30000 nM T43332 C47UEP 11125405 IC50 = 340 nM T43332 CD71SV 11125697 IC50 = 1560 nM T43332 C0SG9J 11136398 IC50 = 200 nM T43332 CMX1S2 11146905 IC50 = 240 nM T43332 CWMD96 11146965 IC50 = 700 nM T43332 C1NMK4 11146971 IC50 = 1530 nM T43332 C5KG1A 11164549 Ki = 35 nM T43332 CR0S7Z 11188883 Ki = 1510 nM T43332 CLA93S 11237163 Ki > 16000 nM T43332 CQFP08 11273559 Ki = 124 nM T43332 CB5RC4 11274304 Ki = 90 nM T43332 CR8NW9 11351302 Ki > 10000 nM T43332 C8WZ0P 11416498 Ki = 430 nM T43332 CVI82D 11479420 Ki > 15000 nM T43332 CK34OX 11509611 Ki > 10900 nM T43332 CO68MA 11524737 Ki > 10900 nM T43332 CWNA56 11621154 IC50 = 6.2 nM T43332 C7EY5G 11654059 Ki = 520 nM T43332 CJP9O1 11684611 Ki = 4220 nM T43332 CL8HU6 11730709 IC50 = 25000 nM T43332 CNZ04Q 11740591 Ki > 15000 nM T43332 C8GJO7 11754872 IC50 > 33000 nM T43332 COM9B5 11763170 IC50 > 30000 nM T43332 C8INH6 11814686 IC50 = 17800 nM T43332 CYX74A 11824584 Ki = 5500 nM T43332 C79MQD 11826825 IC50 > 30000 nM T43332 C61GPA 11828451 IC50 = 1030 nM T43332 CW6E7I 11828640 IC50 = 90 nM T43332 C5SEB3 11967063 IC50 = 5600 nM T43332 CTB2C9 11967128 IC50 = 760 nM T43332 CT7IR8 12110710 IC50 > 100000 nM T43332 CX1ZD7 15521687 Ki = 20900 nM T43332 C60JFG 15521694 Ki = 970 nM T43332 C7VH6K 15950345 Ki > 15000 nM T43332 C3LD4S 16037830 Ki = 13 nM T43332 C53YRO 16098910 IC50 = 38000 nM T43332 C43UDK 20608737 IC50 > 30000 nM T43332 CW3I9O 20608738 IC50 > 30000 nM T43332 C4UZO0 20608741 IC50 = 12500 nM T43332 C9Z2VH 20608755 IC50 > 30000 nM T43332 C3OF2S 20608756 IC50 = 12000 nM T43332 CMX4Q6 20608776 IC50 = 3000 nM T43332 CZ6KH9 20760195 Ki > 15000 nM T43332 CGD57F 20802932 IC50 > 30000 nM T43332 CO2FM4 20802944 IC50 = 26800 nM T43332 C1P0WC 20802959 IC50 = 30000 nM T43332 CBL6N1 20802966 IC50 = 10700 nM T43332 C58KLE 20802993 IC50 = 52 nM T43332 C27ZJT 20802995 IC50 = 7020 nM T43332 CKT23G 22125586 Ki = 900 nM T43332 CV92DP 22351285 Ki = 1 nM T43332 CUXK90 22628841 Ki = 39000 nM T43332 CTFD03 22713561 Ki = 2170 nM T43332 CSJF79 22713564 Ki = 730 nM T43332 CNU61C 22713567 Ki = 1940 nM T43332 C4W0GT 22713568 Ki = 26 nM T43332 C9VHX4 22713571 Ki = 3940 nM T43332 C3VZ7S 23283289 Ki = 40 nM T43332 CV5NL8 23283331 Ki = 350 nM T43332 CRX19I 23646295 Ki > 15000 nM T43332 CQB29J 23646453 Ki = 190 nM T43332 CSY57G 23646463 Ki = 160 nM T43332 CG3W5Q 23661706 IC50 = 60 nM T43332 CKH4O5 24180463 Ki > 11000 nM T43332 CJ3FB7 24871841 Ki = 91 nM T43332 CI8HE3 25138142 IC50 > 33000 nM T43332 C2H4PJ 25166809 Ki > 13000 nM T43332 CR87PA 25171674 Ki = 360 nM T43332 CVU1T9 44277085 IC50 = 4300 nM T43332 C19OGX 44278104 Ki = 140 nM T43332 C3NV7U 44282138 Ki = 31000 nM T43332 C4A1ZJ 44282153 Ki = 27 nM T43332 C5Z6HO 44282567 Ki = 540 nM T43332 CC85WL 44282600 Ki = 45800 nM T43332 C5DZ4L 44282601 Ki = 67 nM T43332 CW9YJ5 44282616 Ki = 3760 nM T43332 CAT3F6 44282630 Ki = 120 nM T43332 C27UQM 44282677 Ki = 3200 nM T43332 CRT93X 44282678 Ki = 7620 nM T43332 CA6X2L 44283195 Ki = 20200 nM T43332 C9IN4E 44314967 IC50 = 290 nM T43332 CVR6K0 44330453 IC50 = 1100 nM T43332 C5W1DZ 44330605 IC50 = 4600 nM T43332 C76ZOE 44330607 IC50 = 109000 nM T43332 C6B0DP 44330620 IC50 = 420 nM T43332 CI8U6O 44338109 IC50 = 706 nM T43332 C9WR3T 44338140 IC50 = 8500 nM T43332 CZW8I0 44338156 IC50 = 22000 nM T43332 C7KM8P 44338170 IC50 > 25000 nM T43332 CUD4G3 44338355 IC50 > 25000 nM T43332 CRMU28 44338377 IC50 = 25000 nM T43332 CV8FM3 44338378 IC50 = 18000 nM T43332 C3F0GD 44338380 IC50 > 25000 nM T43332 CA1G6Q 44338381 IC50 > 25000 nM T43332 CDMG63 44347916 Ki = 47 nM T43332 CEP6C1 44347929 Ki = 20 nM T43332 CC50UP 44347950 Ki = 30 nM T43332 C0PR3S 44347951 Ki = 34 nM T43332 CW2B1L 44347973 Ki = 142 nM T43332 CKBN18 44348006 Ki = 20 nM T43332 CX85LK 44348013 Ki = 156 nM T43332 CQTB91 44348014 Ki = 26 nM T43332 CIB29S 44348020 Ki = 190 nM T43332 CXN6O9 44348021 Ki = 78 nM T43332 C64JUL 44348030 Ki = 43 nM T43332 CPV7C4 44348111 Ki = 33 nM T43332 CTW18J 44348126 Ki = 133 nM T43332 C4G1JX 44348138 Ki = 7000 nM T43332 CO5Y7S 44348145 Ki = 15 nM T43332 C6O8NQ 44348177 Ki = 196 nM T43332 CQM0O4 44348226 Ki = 23 nM T43332 CT09HX 44348227 Ki = 483 nM T43332 CPD32J 44348228 Ki = 83 nM T43332 C9QI8B 44348229 Ki = 256 nM T43332 CWQT21 44348232 Ki = 77 nM T43332 CQA84Y 44386555 Ki = 470 nM T43332 C6SV1C 44387258 IC50 = 35000 nM T43332 CN2GR5 44390800 Ki = 2 nM T43332 CW3G5V 44390801 Ki = 7 nM T43332 CL8T5R 44399322 IC50 = 12 nM T43332 C7GVD8 44399323 IC50 = 20 nM T43332 C18QEF 44399324 IC50 = 21 nM T43332 CLQ92N 44399325 IC50 = 23 nM T43332 CH5YM4 44399326 IC50 = 152 nM T43332 C68ASU 44399327 IC50 = 1.7 nM T43332 CH9TP3 44402039 Ki = 783 nM T43332 C49CME 44402191 Ki = 646 nM T43332 CL80DH 44402364 Ki = 133 nM T43332 CQ4J2A 44402383 Ki = 305 nM T43332 C8WR3I 44402428 Ki = 142 nM T43332 CJQ8X6 44402429 Ki = 195 nM T43332 C6CZ8H 44402442 Ki = 1312 nM T43332 CPLF17 44402521 Ki = 121 nM T43332 C5JK1T 44402528 Ki = 282 nM T43332 C9CWT3 44402591 Ki = 194 nM T43332 CV0S6N 44402617 Ki = 207 nM T43332 C1G4BC 44407625 Ki = 460 nM T43332 C3BX5Y 44412781 Ki > 150000 nM T43332 CCDB58 44413704 Ki = 120 nM T43332 CYLU35 44413709 Ki = 16 nM T43332 CZOF13 44413710 Ki = 17 nM T43332 CGJ80A 44413801 Ki = 3 nM T43332 CO8A0Y 44414333 Ki = 140000 nM T43332 CGV1I0 44426657 IC50 = 20 nM T43332 CXI16J 44426658 IC50 = 40 nM T43332 CZ9O0J 44426660 IC50 = 5480 nM T43332 CJN3M1 44426799 IC50 = 790 nM T43332 CO9Q4B 44427316 IC50 > 30000 nM T43332 CD9O6E 44427319 IC50 > 30000 nM T43332 CVO5Q1 44432538 Ki > 10000 nM T43332 CR16BF 44434808 Ki > 11000 nM T43332 CQIX73 44434809 Ki > 11000 nM T43332 C5R8HJ 44434815 Ki > 11000 nM T43332 COG34X 44434818 Ki > 11000 nM T43332 C9T1DP 44434835 Ki > 11000 nM T43332 CN65UR 44453506 IC50 = 300 nM T43332 CVZW52 44537923 IC50 = 51000 nM T43332 C0PMW3 44584374 Ki = 1320 nM T43332 CR6X5Q 44587208 Ki = 69 nM T43332 C87KXE 44587209 Ki = 25 nM T43332 C94YMX 44587229 Ki = 198 nM T43332 C09ROK 44587230 Ki = 114 nM T43332 CGOR19 44587231 Ki = 35 nM T43332 C8WH9R 44587232 Ki = 15 nM T43332 C3WOP7 44587261 Ki = 130 nM T43332 CX1DP6 44587262 Ki = 42 nM T43332 C7K6JN 44587263 Ki = 43 nM T43332 CKL1J2 44587264 Ki = 18 nM T43332 CTF79D 44587290 Ki = 35 nM T43332 CBXY02 44587291 Ki = 74 nM T43332 CDBV80 44587292 Ki = 30 nM T43332 CWZ34J 44587314 Ki = 20 nM T43332 CI51KQ 44587315 IC50 = 2400 nM T43332 C1LR3H 44587316 IC50 = 6000 nM T43332 CN2A1O 44587317 IC50 = 5000 nM T43332 C2PVE0 45103523 Ki > 26000 nM T43332 CGN14R 45103723 Ki > 26000 nM T43332 CUQF60 45261201 IC50 > 10000 nM T43332 CEXO72 45261244 IC50 = 520 nM T43332 C0H3UO 46878241 Ki = 1011 nM T43332 CNVR31 46905372 IC50 = 1600 nM T43332 CA6GQ5 53341037 Ki = 3190 nM T43332 CV60BK 53488415 Ki = 3684 nM T43332 C9YXM2 56659587 IC50 > 1340000 nM T43332 C2T1WM 56665604 IC50 = 300 nM T43332 CMG9H6 56666511 IC50 > 580000 nM T43332 C0M3AE 56673432 IC50 > 1480000 nM T43332 CI6RX7 56673433 IC50 = 26000 nM T43332 C7DE8I 56676739 IC50 > 1340000 nM T43332 CE4AT6 56676740 IC50 > 400000 nM T43332 C8CN9W 56676741 Ki = 8000 nM T43332 C5LVJ2 56680051 IC50 = 640000 nM T43332 CKF2M0 56680052 Ki = 89000 nM T43332 CJ5SA4 57803617 Ki = 49 nM T43332 C07FPO 57803627 Ki = 1100 nM T43332 C63FQC 57803696 Ki = 10 nM T43332 C5FD3R 57803704 Ki = 750 nM T43332 CLV91D 57803729 Ki = 13 nM T43332 CEH39Z 57803776 Ki = 1.7 nM T43332 C2W7GY 57803799 Ki = 48 nM T43332 C1BZS8 57803813 Ki = 420 nM T43332 CN1HL9 57803827 Ki = 80 nM T43332 C3PV0I 57803829 Ki = 2100 nM T43332 CU4N3X 57803861 Ki = 19 nM T43332 CEG27C 57803875 Ki = 37 nM T43332 C8J7OW 57803884 Ki = 140 nM T43332 CI6U8B 57803906 Ki = 11 nM T43332 CT7RP1 57803917 Ki = 49 nM T43332 C6X3ER 57803948 Ki = 1020 nM T43332 CH2QT8 57804013 Ki = 5 nM T43332 C45OXB 57804023 Ki = 6.1 nM T43332 C37DJW 57804045 Ki = 79 nM T43332 C9EJ7H 57804057 Ki = 68 nM T43332 C7WYV9 57804066 Ki = 20 nM T43332 CFMO72 57804069 Ki = 207 nM T43332 CWJL97 57842563 Ki = 9200 nM T43332 CW0TZ2 57842686 Ki = 2100 nM T43332 C9XW1C 57842830 Ki = 23 nM T43332 CO2IQ4 57842911 Ki = 940 nM T43332 C60HCV 57976401 Ki > 13400 nM T43332 CHB27Y 57976410 Ki > 13390 nM T43332 CM8UJ7 57976444 Ki > 13000 nM T43332 CQ71KE 57976446 Ki > 13000 nM T43332 C91APY 59095797 IC50 = 7 nM T43332 C40NCE 59095829 IC50 = 23 nM T43332 C69SED 59095888 IC50 = 13 nM T43332 CRA2I8 59095906 IC50 = 101 nM T43332 CYB84G 59095944 IC50 = 11 nM T43332 CVP7D6 59315129 Ki = 1500 nM T43332 CI2X9L 59315479 Ki = 9.6 nM T43332 CPW2H7 59315536 Ki = 4.2 nM T43332 CO38AC 59402011 Ki > 13000 nM T43332 C7IO5P 60150643 Ki = 15000 nM T43332 C6JP8Q 60154989 Ki = 630 nM T43332 CWCA65 66573845 IC50 > 1000000 nM T43332 C3LT2W 66674079 Ki > 10900 nM T43332 C23QOJ 66674821 Ki > 10900 nM T43332 CWOD93 66744646 Ki = 1670 nM T43332 C91QMH 68814251 Ki = 1800 nM T43332 CYL98H 68815937 Ki = 15 nM T43332 CA5DG8 69249482 Ki = 1.9 nM T43332 C6AU1R 70252985 Ki > 13300 nM T43332 CTO5I6 70253788 Ki > 13300 nM T43332 C0BPW3 70290375 Ki = 840 nM T43332 C9EL3C 71260387 Ki > 13300 nM T43332 CJPF90 71548883 Ki > 13000 nM T43332 C53BYN 71580813 Ki = 0.62 nM T43332 C57PCL 71580892 Ki = 8.1 nM T43332 CRD4I9 71625797 Ki > 15000 nM T43332 C62ZTJ 71660643 IC50 = 175 nM T43332 C78DJQ 71711730 IC50 < 10000 nM T43332 C4TP1M 71748092 Ki = 15000 nM T43332 CVM7Y6 71748093 Ki = 15000 nM T43332 C8HZ6Q 71748094 Ki = 15000 nM T43332 C6CB0G 71748095 Ki = 15000 nM T43332 C2Z7XJ 71748113 Ki = 15000 nM T43332 C02DQB 72163853 IC50 = 12.5 nM T43332 C3DWZ2 72163854 IC50 = 111 nM T43332 CH6NJ7 72163855 IC50 = 34 nM T43332 C29WAT 72163856 IC50 = 113 nM T43332 C1GI7K 72163964 IC50 = 437 nM T43332 CQ8Y6X 72163965 IC50 = 357 nM T43332 C7IQ6M 72163966 IC50 = 499 nM T43332 CE7P1L 72163967 IC50 = 51 nM T43332 CPDW92 72164078 IC50 = 9 nM T43332 CRBH34 72164200 IC50 = 60 nM T43332 CWNZ45 72164201 IC50 = 164 nM T43332 C0TH5C 72164202 IC50 = 265 nM T43332 CW3QR2 72712049 Ki > 250000 nM T43332 CAL2W7 72712050 Ki > 250000 nM T43332 C2A4TH 72712051 Ki > 250000 nM T43332 CN73TI 72712053 Ki > 250000 nM T43332 C3J8RV 72712070 Ki > 250000 nM T43332 CAZ5R4 72725806 Ki = 280 nM T43332 CPW7T3 72725807 Ki = 41 nM T43332 C4FQ0W 73345765 Ki = 1900 nM T43332 CCD54H 73345766 Ki > 3000 nM T43332 CO4A1M 73345767 Ki > 14000 nM T43332 CC2FW1 73345771 Ki = 14000 nM T43332 C3O9CW 73346025 Ki = 1800 nM T43332 CQGI64 73347555 Ki = 8800 nM T43332 CQF46R 73348759 Ki > 3000 nM T43332 CJG30R 73348764 Ki = 2600 nM T43332 CUD26E 73348765 Ki = 7160 nM T43332 CSQ41U 73348767 Ki > 3000 nM T43332 C82ALB 73350260 IC50 = 1.9 nM T43332 CHF47P 73350338 Ki = 3940 nM T43332 C5VP6W 73350339 Ki = 2400 nM T43332 CK45HD 73350340 Ki = 3000 nM T43332 C60BNQ 73350342 Ki > 3000 nM T43332 CPVC67 73351762 IC50 = 3.4 nM T43332 C2NEV3 73351853 Ki = 7700 nM T43332 CX1WJ7 73351856 Ki = 1500 nM T43332 C4CD7U 73351857 Ki = 2700 nM T43332 C69BHN 73353326 Ki > 3000 nM T43332 C26QPS 73353327 Ki = 1400 nM T43332 C7DGZ9 73353328 Ki = 2500 nM T43332 CA2P1B 73353330 Ki = 2200 nM T43332 CS7FH0 73354754 IC50 = 2.4 nM T43332 COF2K0 73354849 Ki > 3000 nM T43332 C3VFD6 73354850 Ki > 3000 nM T43332 CL34CV 73354863 Ki = 4200 nM T43332 C8N4RM 73356390 Ki = 2100 nM T43332 CH1BJ2 76311085 Ki = 290 nM T43332 C9OKI1 76311087 Ki = 451 nM T43332 CZU72O 76311088 Ki = 275 nM T43332 CE3ZI8 76311089 Ki = 3060 nM T43332 C29QNE 76311090 Ki = 1960 nM T43332 C3R8LG 76311091 Ki = 56 nM T43332 CSBD17 76314701 Ki = 705 nM T43332 CSY3T8 76318271 Ki = 2200 nM T43332 CI7MO1 76318272 Ki = 237 nM T43332 C28QGR 76318273 Ki = 1290 nM T43332 C4WUP1 76318274 Ki = 16300 nM T43332 C9PJ1H 76321975 Ki = 867 nM T43332 C7UP8I 76321976 Ki = 520 nM T43332 CHNJ05 76325595 Ki = 95 nM T43332 C6UR1G 76325596 Ki = 25 nM T43332 C3W5PN 76329159 Ki = 2600 nM T43332 CJ9D8H 76329160 Ki = 474 nM T43332 C6CW8M 76332426 Ki > 100000 nM T43332 CL09IJ 76332819 Ki = 89 nM T43332 CXKG18 76332820 Ki = 610 nM T43332 CYCA26 76332821 Ki = 450 nM T43332 CADC95 76336441 Ki = 442 nM T43332 CZ4N5I 76336442 Ki = 1770 nM T43332 C7TNX2 76336443 Ki = 230 nM T43332 CAT95V 76685067 IC50 > 100000 nM T43332 CMD5V7 86583041 Ki > 10890 nM T43332 CO6U9I 88582319 Ki > 13300 nM T43332 COH41Y 91666660 Ki = 1100 nM T43332 CKS29X 118713018 IC50 > 100000 nM T43332 CRF62H 118713026 IC50 > 100000 nM T43332 CAS3L5 118713029 IC50 > 100000 nM T43332 C3MVG0 118720988 Ki > 10900 nM T43332 C9M2IH 118720990 Ki > 10900 nM T43332 C1E6GW 118720991 Ki > 10900 nM T43332 C9BVI5 118720993 Ki > 10900 nM T43332 C1FQZ6 118720994 Ki > 10900 nM T43332 C0WZA2 118720996 Ki > 10900 nM T43332 CE89KB 118720997 Ki > 10900 nM T43332 CIAL50 118720998 Ki > 10900 nM T43332 C4HLM3 118720999 Ki > 10900 nM T43332 CLD6I3 118721000 Ki > 10900 nM T43332 C0XG7H 118721001 Ki > 10900 nM T43332 CZC53M 118721002 Ki > 10900 nM T43332 C8FZ2L 118721003 Ki > 10900 nM T43332 C0M4IQ 118721004 Ki > 10900 nM T43332 CLRB29 118721005 Ki > 13390 nM T43332 C9B1FX 118721007 Ki > 10900 nM T43332 CRV5Y1 118721008 Ki = 4220 nM T43332 CH6AQ9 118721009 Ki = 6200 nM T43332 CHQ5P7 118987013 Ki > 12170 nM T43332 CK0W2P 127027635 Ki > 13000 nM T43332 CPC0M8 127031390 Ki > 15180 nM T43332 C85ROH 127041472 IC50 > 100000 nM T43332 C7H4XJ 135415880 Ki = 9 nM T43332 C2I6WX 135430716 Ki = 15 nM T43332 C8U2TW 135430841 Ki = 50 nM T43332 C5Q9GO 135430914 Ki = 22 nM T43332 CHMD42 135431470 Ki = 300 nM T43332 CNZ53U 135450094 Ki = 12 nM T43332 CG8Z6V 135450117 Ki = 280 nM T43332 CI40AR 135450152 Ki = 25 nM T43332 CH89OV 135450153 Ki = 14 nM T43332 CPK1H2 135450157 Ki = 1 nM T43332 C4M5BF 135450980 Ki > 75000 nM T43332 CX62AU 135453491 Ki = 135 nM T43332 C6SRC3 135453508 Ki = 730 nM T43332 CTSY50 135453509 Ki = 21 nM T43332 C0UC7X 135453511 Ki = 68 nM T43332 C9WK1B 135456049 Ki = 120 nM T43332 CM7S1D 135457527 Ki = 5 nM T43332 CT27VM 135490247 Ki = 20 nM T43332 C9DRQ8 135528469 Ki = 5.4 nM T43332 CSW47P 135528873 Ki = 14 nM T43332 CYJ02B 135530536 Ki = 13 nM T43332 CQ3YN8 135530560 Ki = 4 nM T43332 C8XC5J 135530568 Ki = 33 nM T43332 CBA90J 135532848 Ki = 38 nM T43332 CR6B1G 135532849 Ki = 500 nM T43332 CZHK63 135532851 Ki = 88 nM T43332 CW6DR2 135543006 Ki = 77 nM T43332 C8G4XP 135543032 Ki = 4000 nM T43332 C3L7ZH 135543057 Ki = 6 nM T43332 CE12AK 135547881 Ki = 10 nM T43332 C7Q9YK 135559071 Ki = 11000 nM T43332 CAU8S4 135559072 Ki = 39000 nM T43332 CXYK80 135559073 Ki = 2400 nM T43332 CA8Q5B 135559074 Ki = 7400 nM T43332 CJNV82 135559075 Ki = 2500 nM T43332 C0HK1X 135559076 Ki = 12000 nM T43332 C2KT9Y 135559077 Ki = 62 nM T43332 C96UQZ 135559078 Ki = 1400 nM T43332 CTM4S0 135559104 Ki = 74 nM T43332 CZPS79 135559105 Ki = 22 nM T43332 C0KE3U 135559106 Ki = 27 nM T43332 C57BFN 135559107 Ki = 29 nM T43332 CF8LZ7 135559108 Ki = 36 nM T43332 C3N1HW 135559111 Ki = 66 nM T43332 CI8CE9 135559112 Ki = 76 nM T43332 CLO7N0 135559114 Ki = 110 nM T43332 CSW10A 135559115 Ki = 130 nM T43332 CYD5H1 135559116 Ki = 120 nM T43332 CMQP13 135559118 Ki = 210 nM T43332 CWE1Q5 135559119 Ki = 250 nM T43332 CGL3D0 135559120 Ki = 270 nM T43332 CVOC19 135559122 Ki = 330 nM T43332 CRE82I 135559123 Ki = 420 nM T43332 CD8XW3 135559124 Ki = 420 nM T43332 CZQ79E 135559125 Ki = 440 nM T43332 CB5H2U 135559126 Ki = 550 nM T43332 CFU9X3 135559127 Ki = 780 nM T43332 C90YUE 135559128 Ki = 880 nM T43332 C5DQ1E 135559129 Ki = 2250 nM T43332 C1T9HA 135559130 Ki = 6400 nM T43332 C1QWR8 135559131 Ki = 16000 nM T43332 C9WN7U 136043834 Ki = 14 nM T43332 CQ9OC5 136043835 Ki = 4 nM T43332 CDGY58 136094842 Ki = 37000 nM T43332 C6FIP1 136094843 Ki = 410 nM T43332 CQW40T 136104458 IC50 = 190 nM T43332 CI7XJ3 136104459 IC50 = 110 nM T43332 CPI6G8 136106132 Ki = 54 nM T43332 C2W0KO 136106133 Ki = 64 nM T43332 CDQ62V 137637214 Ki > 50000 nM T43332 C2K8JV 137639385 Ki > 50000 nM T43332 CA8E9H 137650038 Ki = 61 nM T43332 CX4F8N 137650590 Ki > 10000 nM T43332 CNX46H 137654508 Ki > 50000 nM T43332 CX07YE 139592452 Ki = 4850 nM T43332 CE6C0A 145970642 Ki = 3280 nM T43332 CICU31 155511394 Ki = 7995 nM T43332 C2VX3G 155512946 Ki > 13300 nM T43332 C2CI8S 155513907 Ki = 11574 nM T43332 C37MUL 155515203 IC50 = 12 nM T43332 C3AL6D 155533619 IC50 = 11 nM T43332 CY3FE6 155533938 IC50 = 4.7 nM T43332 D02KKL 1282 Ki = 74 nM T43332 D02XPB 23646462 Ki = 1000 nM T43332 D0CT8A 23646461 Ki = 4200 nM T43332 D0JU9N 6914623 Ki > 2800 nM T43332 D0K7YL 447476 Ki = 160 nM T43332 D0ON2Z 204102 Ki > 2300 nM T43332 D0V7RD 10439038 Ki = 108 nM T55435 CV9X6A 385917 Ki = 3860 nM T55435 CUG5J1 9901007 IC50 = 1350 nM T55435 CBEX76 10268287 IC50 = 440 nM T55435 CCK69R 11252976 IC50 = 20000 nM T55435 C16OWH 12594528 Ki = 7320 nM T55435 CO31XL 14203721 Ki = 22870 nM T55435 C67JBF 14203722 Ki = 12480 nM T55435 C9UZ4P 14203723 Ki = 10790 nM T55435 CZ9G5K 25238874 Ki = 9210 nM T55435 CWM7N0 25239176 Ki = 3530 nM T55435 CSCZ56 46898076 IC50 = 176 nM T55435 CKO8C1 50898364 Ki < 1.3 nM T55435 C2NA0G 50943292 Ki = 17 nM T55435 CN13QO 50943377 Ki = 4 nM T55435 CZYP20 50943452 Ki < 1 nM T55435 CYN94V 50943864 Ki = 4 nM T55435 CH7U3Q 56956255 IC50 = 40 nM T55435 CIZ59T 58169162 Ki = 13 nM T55435 CWJ26R 60150737 IC50 = 23 nM T55435 CRL57E 68375232 Ki > 4000 nM T55435 C9NMO5 70681209 IC50 = 223 nM T55435 CF4XW9 70681210 IC50 = 393 nM T55435 C53AXH 70681211 IC50 = 241 nM T55435 C9I7WP 70681212 IC50 = 1130 nM T55435 CH76ZU 70683296 IC50 = 375 nM T55435 CDU16I 70683297 IC50 = 354 nM T55435 C5ER7B 70683298 IC50 = 56 nM T55435 CR1HC4 70685404 IC50 = 87 nM T55435 CD26IT 70685405 IC50 = 88 nM T55435 CR1I7X 70685406 IC50 = 1990 nM T55435 CW7Z6X 70687546 IC50 = 1162 nM T55435 C2OI8P 70687547 IC50 = 107 nM T55435 CKG4D8 70687548 IC50 = 53 nM T55435 C7ZN4E 70689605 IC50 = 384 nM T55435 CX6F0N 70689606 IC50 = 202 nM T55435 CL7H9A 70689607 IC50 = 84 nM T55435 CL31BP 70689608 IC50 = 217 nM T55435 COVX36 70689609 IC50 = 115 nM T55435 CB39HO 70689610 IC50 = 73 nM T55435 C3K7JC 70689611 IC50 = 56 nM T55435 CRT10E 70691734 IC50 = 74 nM T55435 C50QZV 70691735 IC50 = 64 nM T55435 C2C1FA 70693802 IC50 = 322 nM T55435 C89SXK 70693803 IC50 = 453 nM T55435 CC0L4W 70693804 IC50 = 428 nM T55435 CVYG19 70693805 IC50 = 39 nM T55435 CDSA05 70693806 IC50 = 40 nM T55435 C14QZG 70695925 IC50 = 86 nM T55435 CR35AQ 70695926 IC50 = 715 nM T55435 CC9JO6 70695927 IC50 = 121 nM T55435 C0I5YK 70695928 IC50 = 55 nM T55435 CNJQ63 118715295 Ki = 6380 nM T55435 C9QK3E 118715296 Ki = 7680 nM T55435 CJ3RB1 118715297 Ki = 7010 nM T55435 CSPR50 118715298 Ki = 5250 nM T55435 CKRC59 118715299 Ki = 13130 nM T55435 CXN61W 118715300 Ki = 26510 nM T55435 CKI3E0 118715301 Ki = 9040 nM T55435 C5JTE2 118715302 Ki = 7590 nM T55435 CFX51G 118715303 Ki = 18460 nM T55435 C57VKN 134815860 Ki < 2 nM T55435 CW3P2E 134815875 Ki < 1 nM T55435 C6X4LW 134816069 Ki = 46 nM T55435 CK7RY6 134816070 Ki = 40 nM T55435 CK4PN9 134816385 Ki = 38 nM T55435 C9H7YQ 134816426 Ki = 960 nM T55435 CSJ1V7 134816427 Ki = 150 nM T55435 C4F6CH 134816428 Ki = 230 nM T55435 CSZM60 134816433 Ki = 50 nM T55435 CNI8R2 134816434 Ki = 15 nM T55435 CUVZ68 134816435 Ki = 23 nM T55435 CWM89T 134816436 Ki = 23 nM T55435 C98PFY 134816472 Ki = 82 nM T55435 CO05YI 134816473 Ki = 150 nM T55435 CX2GT5 134816476 Ki = 190 nM T55435 C21ZPH 134816477 Ki = 310 nM T55435 CE01BG 134816532 Ki = 29 nM T55435 CNK2R8 134816533 Ki = 88 nM T55435 CBH0E8 134816534 Ki = 24 nM T55435 CRT3W9 134816535 Ki = 6 nM T55435 CH7VQ4 134816642 Ki = 150 nM T55435 CK65PU 134816643 Ki = 81 nM T55435 CB7OG9 134816644 Ki = 98 nM T55435 C0OX5I 134816676 Ki = 990 nM T55435 C0N4GD 134816677 Ki = 1400 nM T55435 C5I0ZM 134816678 Ki = 310 nM T55435 CWZL67 134816679 Ki = 72 nM T55435 C2Z6OV 134816680 Ki = 60 nM T55435 C5OW3X 134816681 Ki = 5 nM T55654 D05LYX 3488 IC50 = 15000 nM T55654 D0W7WC 16220172 EC50 = 3 nM T55654 D0E0JO 117857370 EC50 = 181 nM T55654 D0X0CB 16678941 EC50 = 2570.4 nM T55654 CDVF74 386896 EC50 = 146000 nM T55654 CS3W5K 679184 EC50 = 200 nM T55654 C1XP4H 723141 EC50 > 10000 nM T55654 CGR03J 1144671 EC50 = 1096.48 nM T55654 CQ0PH4 1206778 EC50 = 2100 nM T55654 CXW45L 1207558 IC50 = 30000 nM T55654 CHZP28 1320951 IC50 = 1500 nM T55654 CZW62F 1381792 EC50 = 240 nM T55654 CRTC48 1554208 IC50 = 300 nM T55654 CT9LF0 1554549 IC50 = 7000 nM T55654 C9TLR2 1608007 IC50 = 28000 nM T55654 CT6HO1 1640986 EC50 = 7900 nM T55654 C4FEK0 1776674 IC50 = 2600 nM T55654 CA3LH9 2046483 IC50 = 24000 nM T55654 C2T9IC 2262781 IC50 = 7000 nM T55654 CX8ZE4 2265553 IC50 = 15000 nM T55654 C19AOD 3214072 EC50 = 3800 nM T55654 CHZ82Q 3217019 EC50 = 3800 nM T55654 CXSN85 3217032 EC50 = 3900 nM T55654 C3ECD9 3221675 EC50 = 14000 nM T55654 CB2J4A 3221704 EC50 = 8200 nM T55654 CM52VC 3224090 EC50 = 1500 nM T55654 C8Q7YM 3760412 EC50 = 200 nM T55654 CC59FL 3942679 EC50 = 120 nM T55654 C52FZO 4656456 EC50 = 16000 nM T55654 C6H9EM 6532107 IC50 = 1400 nM T55654 CL47HK 9795307 EC50 = 141000 nM T55654 CS08ZV 9844005 IC50 = 380000 nM T55654 C13OPT 10087442 EC50 = 70500 nM T55654 COXI63 10358736 EC50 = 23500 nM T55654 CPSB31 11155965 EC50 = 6.3 nM T55654 CDC6K2 11167315 EC50 = 26 nM T55654 CYI9N6 11183685 IC50 = 16 nM T55654 CC62DV 11214961 EC50 = 12 nM T55654 C2DNQ5 11232967 EC50 = 20000 nM T55654 C7SM4F 11248737 EC50 = 11 nM T55654 CZCO36 11260275 EC50 = 6 nM T55654 CSWY38 11275309 IC50 = 5 nM T55654 CAUC38 11295426 EC50 = 9.4 nM T55654 CB02DW 11329834 EC50 = 20 nM T55654 CX83YT 11341447 EC50 = 20 nM T55654 C1DMJ4 11370263 EC50 = 48000 nM T55654 CF5WC4 11375102 EC50 = 119 nM T55654 CX4DK3 11432286 EC50 = 3.5 nM T55654 C0MSX1 11466370 EC50 = 15 nM T55654 C8TF4E 11509534 EC50 = 2884.03 nM T55654 CF8L1D 11530695 IC50 = 160000 nM T55654 C4SX3W 11738767 EC50 = 750 nM T55654 CG49UM 11752089 EC50 = 16 nM T55654 CJA2N0 11771615 EC50 = 26000 nM T55654 CI6P7Q 11785682 EC50 = 23 nM T55654 CLF85K 11957831 EC50 = 2187.76 nM T55654 C9EUQ5 11958611 EC50 = 700 nM T55654 CNE69P 13588670 EC50 = 2110 nM T55654 CQ42FD 16016575 IC50 = 1200 nM T55654 CHMB05 16016583 IC50 = 90 nM T55654 C6TOB8 16016605 IC50 = 800 nM T55654 CCD10N 16023364 IC50 = 3900 nM T55654 CL2JY6 17715303 EC50 = 1300 nM T55654 C1IP0A 17715310 EC50 = 800 nM T55654 CUI03O 17715311 EC50 = 200 nM T55654 C9L8YB 20574550 EC50 = 3500 nM T55654 CPY4W2 20873375 IC50 = 3200 nM T55654 CU72RL 20898903 IC50 = 2500 nM T55654 C58GRH 20898912 IC50 = 1500 nM T55654 CB1X4A 20922628 IC50 = 3900 nM T55654 C0B5LO 23614017 IC50 = 4500 nM T55654 CUW7Y3 23614023 IC50 = 2000 nM T55654 CO8U2F 23614043 IC50 = 1700 nM T55654 CU0V3G 23614049 IC50 = 8000 nM T55654 CP2RO3 23614050 IC50 = 2500 nM T55654 CW9O7C 23614053 IC50 = 5000 nM T55654 CA45HX 23614055 IC50 = 3000 nM T55654 C4GT8C 23614057 IC50 = 3000 nM T55654 C2GOE7 23614069 IC50 = 1500 nM T55654 CTAS72 23614521 IC50 = 12000 nM T55654 CF01YH 23614528 IC50 = 14000 nM T55654 CM7C8Z 24747099 EC50 = 10964.78 nM T55654 CHGO25 24858212 EC50 = 100 nM T55654 CH5I9U 24858374 EC50 = 1700 nM T55654 CP2L3K 24858379 EC50 = 3500 nM T55654 C8ABL2 24882564 IC50 = 170000 nM T55654 C2UHN4 25130495 EC50 = 300 nM T55654 CNAK75 25131145 IC50 = 11000 nM T55654 C6DLT0 25205998 EC50 = 300 nM T55654 CX40LF 25265182 IC50 = 4100 nM T55654 CHFA48 30131597 EC50 = 1500 nM T55654 CPO54W 39887958 EC50 = 800 nM T55654 CP14CO 39888551 EC50 = 100 nM T55654 CQM13N 42647973 IC50 = 1700 nM T55654 C2KP1N 43815411 EC50 = 100000 nM T55654 CCRS82 43815487 EC50 = 1500 nM T55654 CAHZ42 43815502 EC50 = 6700 nM T55654 CW5BR7 44237591 IC50 = 1400 nM T55654 CEB2S8 44237643 IC50 = 11000 nM T55654 C0LEY5 44237644 IC50 = 1500 nM T55654 CL1OX7 44237645 IC50 = 15000 nM T55654 CZD38I 44237646 IC50 = 14000 nM T55654 CF1Q8H 44237647 IC50 = 5000 nM T55654 C4NF9J 44237697 IC50 = 9000 nM T55654 CKDM37 44237744 IC50 = 8000 nM T55654 CM9Y6N 44237745 IC50 = 8700 nM T55654 CI1EB5 44237747 IC50 = 8200 nM T55654 CH7QX6 44387641 EC50 = 292 nM T55654 CTZ13M 44387642 EC50 = 314 nM T55654 C9Y1QO 44399794 EC50 = 294 nM T55654 CYUF10 44399846 EC50 = 202 nM T55654 CC79KZ 44400183 EC50 = 51 nM T55654 CNP5C9 44400200 EC50 = 82 nM T55654 CXK41R 44400217 EC50 = 10 nM T55654 CQXS60 44400252 EC50 = 79 nM T55654 CI76MC 44400376 EC50 = 35 nM T55654 C67TWX 44400611 EC50 = 176 nM T55654 CS8CA2 44400633 EC50 = 145 nM T55654 C6E8NP 44400640 EC50 = 420 nM T55654 CFB6T2 44400645 EC50 = 100 nM T55654 CX2JR1 44400647 EC50 = 230 nM T55654 CMA1Y0 44400665 EC50 = 291 nM T55654 CZ1BE0 44400668 EC50 = 268 nM T55654 C4HA5G 44400669 EC50 = 282 nM T55654 C2UXT6 44400678 EC50 = 336 nM T55654 CWC7A0 44400685 EC50 = 66 nM T55654 CQ8FK3 44400688 EC50 = 66 nM T55654 CZE06Q 44400689 EC50 = 71 nM T55654 C5LAW0 44400705 EC50 = 590 nM T55654 CX2W1F 44400713 EC50 = 41 nM T55654 CN9A4O 44400714 EC50 = 202 nM T55654 CV1JE4 44400715 EC50 = 338 nM T55654 C6D9UG 44400719 EC50 = 61 nM T55654 C78ETN 44400725 EC50 = 167 nM T55654 C0JX3S 44400734 EC50 = 160 nM T55654 CKXI37 44400740 EC50 = 394 nM T55654 CM7PU8 44400747 EC50 = 53 nM T55654 C9C1PF 44446497 IC50 = 330000 nM T55654 CN9BV2 44446499 IC50 = 490000 nM T55654 CG5T1I 44460193 IC50 = 15000 nM T55654 C6HQZ9 44561738 IC50 = 11000 nM T55654 CU8V6K 44561740 IC50 = 25000 nM T55654 CR8KJ4 44561741 IC50 = 27000 nM T55654 C6E8OK 44561743 IC50 = 27000 nM T55654 C3SI7G 44561789 IC50 = 28000 nM T55654 CES65N 44561790 IC50 = 32000 nM T55654 CKAF05 44562004 IC50 = 5000 nM T55654 C97KCM 44562056 IC50 = 13000 nM T55654 C6YFB9 44562115 IC50 = 18000 nM T55654 CJ6V3K 44562116 IC50 = 19000 nM T55654 C17EAX 44562117 IC50 = 20000 nM T55654 C1JE9D 44562118 IC50 = 20000 nM T55654 CCP7X6 44562145 IC50 = 25000 nM T55654 CT1Y6B 44562146 IC50 = 28000 nM T55654 CF5VY2 44562147 IC50 = 29000 nM T55654 CNJV54 44562178 IC50 = 50000 nM T55654 C1KST7 44754025 EC50 = 3000 nM T55654 CIJE76 44815033 IC50 = 700 nM T55654 CYI6J9 46220952 EC50 = 8500 nM T55654 CIS60U 46221178 EC50 = 930 nM T55654 C19FEM 46221179 EC50 = 3000 nM T55654 C1X8BE 46221405 EC50 = 3388.44 nM T55654 CC49MF 46221409 EC50 = 750 nM T55654 C1A6OU 46265602 IC50 = 2500 nM T55654 C6PF0H 46265619 IC50 = 100000 nM T55654 CD1MP0 46265620 IC50 = 1200 nM T55654 CRM9A3 46265640 IC50 = 1700 nM T55654 CKF8R0 46265664 IC50 = 2000 nM T55654 C3CSZ8 46265666 IC50 = 800 nM T55654 CPZ2B8 46269474 IC50 = 2000 nM T55654 C84RKE 46871622 EC50 = 1000 nM T55654 C5JXE6 46888150 EC50 = 1000 nM T55654 C8Z9PN 46888193 EC50 = 1000 nM T55654 C51ZNE 46888194 EC50 = 3000 nM T55654 C8XP1Q 46904956 EC50 = 100000 nM T55654 C9S5WO 46904957 EC50 = 100000 nM T55654 CQ1BZ4 46904958 EC50 = 100000 nM T55654 C4OT0E 46904959 EC50 = 100000 nM T55654 CO1H7B 46904960 EC50 = 4570.88 nM T55654 C5N8GZ 46904961 EC50 = 4265.8 nM T55654 CE0OM5 49864304 IC50 = 2000 nM T55654 C9JSC6 53299902 EC50 = 1500 nM T55654 C9PF3K 53382957 EC50 = 3000 nM T55654 C0T6FP 53382958 EC50 = 100000 nM T55654 C27RNI 53382959 EC50 = 2691.53 nM T55654 CZSP84 53382960 EC50 = 7244.36 nM T55654 CGVT02 53382961 EC50 = 4168.69 nM T55654 C61KWY 53382962 EC50 = 2691.53 nM T55654 CZB9G0 53382963 EC50 = 3700 nM T55654 C8KSU7 53387352 IC50 = 8 nM T55654 C9WQE3 53391641 IC50 = 90 nM T55654 CHQR71 53391642 IC50 = 500 nM T55654 C8CK2V 53391643 IC50 = 150 nM T55654 C60HYM 53391644 IC50 = 370 nM T55654 CK3L0Z 53391645 IC50 = 600 nM T55654 CH3G0A 53391741 IC50 = 25 nM T55654 CHN67U 53391742 IC50 = 25 nM T55654 C15GIQ 53391743 IC50 = 170 nM T55654 CUW1F4 53391744 IC50 = 170 nM T55654 CVY72U 53391745 IC50 = 50 nM T55654 C40EJW 53391844 IC50 = 80 nM T55654 CCH3O4 53392785 IC50 = 2000 nM T55654 CW43TV 53392786 IC50 = 1000 nM T55654 CHKZ24 53392869 IC50 = 300 nM T55654 C4NU0F 53392870 IC50 = 1700 nM T55654 CFT7P0 53392871 IC50 = 1700 nM T55654 CZ93WV 53392872 IC50 = 150 nM T55654 C0H4KJ 53392873 IC50 = 90 nM T55654 CAX7K5 53392963 IC50 = 170 nM T55654 CN3H9Y 53392964 IC50 = 350 nM T55654 C17VCY 56954842 EC50 = 100000 nM T55654 CX1BN9 56954960 EC50 = 100000 nM T55654 C15DCS 56954961 EC50 = 100000 nM T55654 COJ1F5 56954962 EC50 = 100000 nM T55654 CJ0LK2 57391159 EC50 = 1400 nM T55654 CH84EA 57396421 EC50 = 1400 nM T55654 CXS7V4 57567300 EC50 = 6900 nM T55654 C7Q0VO 57567320 EC50 = 6000 nM T55654 C7CN1X 57567354 EC50 = 100 nM T55654 C6UI9E 57567374 EC50 = 3 nM T55654 CPO3Y1 57567409 EC50 = 400 nM T55654 C54JMN 58609876 EC50 = 1584.89 nM T55654 CY4C7V 58609893 EC50 = 8128.31 nM T55654 COW6D8 58910531 EC50 = 71000 nM T55654 C74POU 59549575 IC50 = 9200 nM T55654 CVR52H 66554044 EC50 = 4900 nM T55654 CB9I0Z 66554122 EC50 = 140 nM T55654 C0ZOR4 66554123 EC50 = 1600 nM T55654 C6QE7O 66554124 EC50 = 4600 nM T55654 CDF4P6 66674636 EC50 = 5100 nM T55654 C2YC3G 66674857 EC50 = 100 nM T55654 CLCI18 66674872 EC50 = 5600 nM T55654 CWVD76 66674989 EC50 = 200 nM T55654 CD6KG4 66675121 EC50 = 11 nM T55654 CHO7B4 66675151 EC50 = 8500 nM T55654 C06VXY 66675476 EC50 = 400 nM T55654 CQG7E4 66675750 EC50 = 9 nM T55654 CORZ62 66675903 EC50 = 20 nM T55654 C7HYI5 66676193 EC50 = 100 nM T55654 CGKN91 66676209 EC50 = 6400 nM T55654 CY9R8W 66676213 EC50 = 6100 nM T55654 CJ79LQ 68463495 EC50 = 100 nM T55654 CR30UX 71110482 EC50 = 4200 nM T55654 CLS3A7 71655425 IC50 = 4 nM T55654 CN70BI 74015911 IC50 = 6600 nM T55654 C80BVE 74015912 IC50 = 8700 nM T55654 C1N7XV 74015913 IC50 = 2900 nM T55654 C6NHC5 74015914 IC50 = 8300 nM T55654 C6N5KJ 74015915 IC50 = 4500 nM T55654 CEG9I2 74015918 IC50 = 2100 nM T55654 CWN40L 74015919 IC50 = 5200 nM T55654 CQFA34 74015920 IC50 = 900 nM T55654 C1C4QG 74015921 IC50 = 5200 nM T55654 C1KEQ3 87056011 EC50 < 10000 nM T55654 C9DA8R 87101512 EC50 = 3 nM T55654 C1BYV4 87101517 EC50 = 2 nM T55654 CE32XP 90479852 EC50 = 1320 nM T55654 CNU83T 91594409 EC50 = 5000 nM T55654 CVQZ27 91933842 EC50 = 740 nM T55654 CVA70U 113198968 EC50 = 2187.76 nM T55654 C49NTL 117857707 EC50 = 590 nM T55654 C6H2EL 117857738 EC50 = 123 nM T55654 CFAU29 117857780 EC50 = 199 nM T55654 CY5M1V 117857808 EC50 = 981 nM T55654 CDX6L9 117857842 EC50 = 7777 nM T55654 C58GUC 117857867 EC50 = 130 nM T55654 CQ08WV 117857891 EC50 = 421 nM T55654 CAN29F 117858047 EC50 = 162 nM T55654 C6M3JL 117858183 EC50 = 81 nM T55654 C5G1CL 118710751 IC50 = 8900 nM T55654 CD0P7C 118710752 IC50 = 5800 nM T55654 C6O8WH 118710753 IC50 = 6600 nM T55654 CI8PV6 118710754 IC50 = 8800 nM T55654 CN07SI 118710755 IC50 = 4800 nM T55654 C5KZQ4 118710756 IC50 = 6900 nM T55654 C5OE4B 118710757 IC50 = 7200 nM T55654 C7K6BQ 118710758 IC50 = 2200 nM T55654 CJ2F9R 118710759 IC50 = 3600 nM T55654 C2B9QX 118723015 EC50 = 660 nM T55654 C51GXB 118723017 EC50 = 590 nM T55654 CRJK02 121301060 EC50 = 850 nM T55654 C2ONU3 121301160 EC50 = 20000 nM T55654 CFJ19C 121301281 EC50 = 100 nM T55654 C7J6YH 121301288 EC50 = 1340 nM T55654 CI2A5D 121302336 EC50 = 1160 nM T55654 CB1D0R 121302360 EC50 = 260 nM T55654 CF9GU4 122183923 EC50 = 34000 nM T55654 CAL95F 122183926 EC50 = 27000 nM T55654 CNC6M2 122183935 EC50 = 5300 nM T55654 C1HZW6 122183956 EC50 = 6400 nM T55654 CDX18Q 122183961 EC50 = 8500 nM T55654 CT2A0I 122183963 EC50 = 9500 nM T55654 CMC01O 122183965 EC50 = 58000 nM T55654 CZ8M7K 122183968 EC50 = 5700 nM T55654 C6FR5W 122183986 EC50 = 32000 nM T55654 C7XP6M 122184002 EC50 = 14000 nM T55654 C67ITZ 122184012 EC50 = 15000 nM T55654 CE56DG 127039262 EC50 = 891.25 nM T55654 C4DZ2M 127039611 EC50 = 400 nM T55654 C74IRU 127039612 EC50 = 1400 nM T55654 CMH0R4 127039613 EC50 = 2800 nM T55654 CJ85VW 127040294 EC50 = 3090.3 nM T55654 CF81BC 127040295 EC50 = 1500 nM T55654 COM3S5 127040623 EC50 = 100000 nM T55654 C4QMI3 127040944 EC50 = 100000 nM T55654 CHU9G3 127040945 EC50 = 100000 nM T55654 CIX3Y6 127040946 EC50 = 100000 nM T55654 CY8DL5 127040947 EC50 = 100000 nM T55654 C6P3ML 127040948 EC50 = 100000 nM T55654 CRF7O2 127041267 EC50 = 100000 nM T55654 CQ52CZ 127041881 EC50 = 100000 nM T55654 C0DA2K 127041882 EC50 = 398.11 nM T55654 CJ8MA0 127041883 EC50 = 3467.37 nM T55654 CXP09C 127041884 EC50 = 199.53 nM T55654 C45XQI 127041885 EC50 = 2290.87 nM T55654 CST79L 127041886 EC50 = 199.53 nM T55654 CUR89W 127041889 EC50 = 300 nM T55654 CZ1KE2 127042199 EC50 = 100000 nM T55654 C1D6KM 127042200 EC50 = 100000 nM T55654 CS29FB 127042201 EC50 = 300 nM T55654 C8S1GX 127042202 EC50 = 100000 nM T55654 C41VXA 127042856 EC50 = 700 nM T55654 C5Z0HV 127042857 EC50 = 200 nM T55654 CIM9B7 127042858 EC50 = 200 nM T55654 CG39OY 129285899 EC50 = 31 nM T55654 CQW7S0 129285916 EC50 = 900 nM T55654 CQ8L0R 129285924 EC50 = 160 nM T55654 CB3H0G 129285959 EC50 = 2800 nM T55654 CGJ38R 129285968 EC50 = 5400 nM T55654 CL8G2O 129286459 EC50 = 1000 nM T55654 C13YUN 129286476 EC50 > 10000 nM T55654 CHR71F 129286517 EC50 = 55 nM T55654 CEC87Y 129286522 EC50 > 10000 nM T55654 CJW7T0 129286544 EC50 = 9 nM T55654 CKO90T 129286545 EC50 = 820 nM T55654 CEM6K3 129286546 EC50 > 10000 nM T55654 C0D6PX 129286552 EC50 = 177 nM T55654 C9ZXJ2 129286559 EC50 > 10000 nM T55654 C9DR1E 129286560 EC50 > 10000 nM T55654 CR6NA4 129286562 EC50 = 550 nM T55654 CI64LA 129286564 EC50 = 1000 nM T55654 C2E3JG 129286565 EC50 = 330 nM T55654 CKD67M 129286569 EC50 = 18 nM T55654 CO7BN2 129286574 EC50 = 690 nM T55654 C5KGA3 129286577 EC50 = 52 nM T55654 C3PH8K 129286581 EC50 = 1000 nM T55654 C3OI8C 129286582 EC50 = 10 nM T55654 C2W0AO 129286586 EC50 = 1000 nM T55654 CXC2T6 129286594 EC50 = 65 nM T55654 CSW6M2 129286598 EC50 > 10000 nM T55654 CUY48F 129286601 EC50 = 20 nM T55654 CZKP04 129286602 EC50 = 110 nM T55654 CMRG60 129286606 EC50 = 4300 nM T55654 C7HOT4 129286607 EC50 > 10000 nM T55654 C8W7KU 129286611 EC50 = 70 nM T55654 CRK8E3 129286614 EC50 = 760 nM T55654 C2ZT5U 129286615 EC50 > 10000 nM T55654 CAC9X0 129286616 EC50 = 63 nM T55654 CI2E5S 129286617 EC50 > 10000 nM T55654 CSXL19 129298539 EC50 = 9900 nM T55654 C0XEV6 129304807 EC50 = 2800 nM T55654 CNCI72 129304809 EC50 = 200 nM T55654 C5GN8P 129304810 EC50 = 18000 nM T55654 C7EAZ0 129304811 EC50 = 2500 nM T55654 CTL70X 129304812 EC50 = 4800 nM T55654 C67INA 129304813 EC50 = 140 nM T55654 CJD2P6 129304814 EC50 = 1200 nM T55654 C7A6OJ 129304815 EC50 = 700 nM T55654 C6OPA8 129304816 EC50 = 1600 nM T55654 COW96U 129304818 EC50 = 500 nM T55654 CQL67U 129304820 EC50 = 2000 nM T55654 C0BM9U 129304822 EC50 = 900 nM T55654 COWV21 135899519 IC50 = 760 nM T55654 C25BWR 135915324 IC50 = 17000 nM T55654 C8M5EW 137451669 EC50 > 10000 nM T55654 CHZ0B8 137547622 EC50 = 30 nM T55654 CIO4Z2 137547626 EC50 = 150 nM T55654 CS8C6J 137641555 EC50 = 490 nM T55654 CE26WU 137645512 EC50 > 10000 nM T55654 CKN2M4 137657662 EC50 = 236 nM T55654 CYZ7L5 139443337 EC50 = 66 nM T55654 C6BX2U 139443340 EC50 = 105 nM T55654 CR9QY1 140857358 EC50 = 132 nM T55654 CZJV70 140857394 EC50 = 52 nM T55654 CV8JE6 140857431 EC50 = 1130 nM T55654 C4LV8I 140857436 EC50 = 35 nM T55654 CFRU24 140857457 EC50 = 346 nM T55654 CS54DC 140857462 EC50 = 173 nM T55654 CRT40A 140857572 EC50 = 48 nM T55654 C9SB3P 140857617 EC50 = 137 nM T55654 CD8HE9 140857688 EC50 = 150 nM T55654 CINF18 140857761 EC50 = 213 nM T55654 C5GO7R 140857765 EC50 = 222 nM T55654 CYBS95 140857766 EC50 = 247 nM T55654 CN76UH 140857971 EC50 < 1000 nM T55654 CB89SK 140858249 EC50 < 1000 nM T55654 CJ15SL 140858356 EC50 < 1000 nM T55654 C0XF2K 140858456 EC50 < 1000 nM T55654 CGTK25 140858910 EC50 = 1000 nM T55654 C08DUX 140859316 EC50 < 1000 nM T55654 CLO08A 140859344 EC50 < 1000 nM T55654 CR5E6T 140859382 EC50 < 1000 nM T55654 CXV96R 145948310 IC50 = 15 nM T55654 CO8QL9 145949181 EC50 = 3890.45 nM T55654 COG4W2 145949807 EC50 = 1200 nM T55654 CE26MY 145949920 EC50 = 4897.79 nM T55654 CNE4M0 145949941 EC50 = 891.25 nM T55654 C2E5QT 145949985 EC50 = 7943.28 nM T55654 CL31KV 145950120 EC50 > 5000 nM T55654 CVF0J4 145950265 EC50 = 3019.95 nM T55654 CJ61WI 145950772 EC50 = 199.53 nM T55654 C8V4MN 145950835 EC50 = 1800 nM T55654 C3Z7YP 145950968 EC50 = 199.53 nM T55654 CF59BM 145952012 EC50 = 1698.24 nM T55654 C9HG4X 145952712 EC50 < 1000 nM T55654 CU3YW2 145953159 EC50 = 3981.07 nM T55654 CP17VY 145953201 EC50 = 5370.32 nM T55654 C6PX1Y 145953587 EC50 = 933.25 nM T55654 CL1U6V 145954017 EC50 = 2290.87 nM T55654 C7I3JQ 145954179 EC50 = 891.25 nM T55654 C6Q1UG 145954329 EC50 > 5000 nM T55654 CRM93L 145954588 EC50 = 1000 nM T55654 CLHX06 145954898 EC50 = 8511.38 nM T55654 CN76CT 145954901 EC50 = 3019.95 nM T55654 C79LGY 145956272 EC50 = 300 nM T55654 CP48NT 145957156 EC50 = 2290.87 nM T55654 CU12HF 145957495 EC50 = 2884.03 nM T55654 CFOX47 145958109 EC50 = 549.54 nM T55654 CI86RA 145958124 EC50 = 3800 nM T55654 COB0D3 145958847 EC50 = 1200 nM T55654 CQ4P1V 145959265 EC50 = 2089.3 nM T55654 CSMU43 145959988 EC50 = 2884.03 nM T55654 C1SJ7R 145960012 EC50 = 1288.25 nM T55654 CETC71 145960137 EC50 = 1000 nM T55654 CZ67KO 145960998 EC50 = 87 nM T55654 CSEK64 145961627 EC50 = 758.58 nM T55654 C2GU4L 145974102 EC50 = 1900 nM T55654 CPO2Q8 145985497 IC50 = 58620 nM T55654 C38APU 146013863 EC50 = 0.5 nM T55654 C4P3ZQ 155512929 EC50 = 2010 nM T55654 C1Q7US 155516088 EC50 = 1400 nM T55654 CA7H6F 155542938 EC50 = 1970 nM T55654 D00RIX 5280443 EC50 = 9000 nM T55654 D02XHC 448912 EC50 = 111 nM T55654 D0S1FV 135476586 IC50 = 5000 nM T72267 D0O3OS 104850 EC50 = 10100 nM T72267 D0P1FO 16078 EC50 = 960 nM T72267 CVL1A0 320263 IC50 > 10000 nM T72267 CL3UD5 320264 IC50 > 10000 nM T72267 CFY02L 356017 IC50 > 10000 nM T72267 C8X7ST 356018 IC50 > 10000 nM T72267 CGT6F3 738959 IC50 > 10000 nM T72267 C0MYU2 1281700 IC50 > 10000 nM T72267 C8KD9F 1281702 IC50 > 10000 nM T72267 CH8PY0 1281704 IC50 > 10000 nM T72267 CX5F6G 1281706 IC50 = 10000 nM T72267 CC4B0K 5917569 IC50 > 10000 nM T72267 C1RO9M 9887568 IC50 > 10000 nM T72267 C73TBN 10468802 IC50 > 10000 nM T72267 C8LF3D 10858553 IC50 > 10000 nM T72267 C3TC7H 10871668 IC50 = 33000 nM T72267 CSG5H6 10902223 IC50 > 10000 nM T72267 CCI2L6 11045217 IC50 > 10000 nM T72267 CI8A6B 11076506 IC50 > 10000 nM T72267 C9E2AP 11152300 IC50 = 14100 nM T72267 C92AOP 11187538 IC50 > 10000 nM T72267 CYE8Q0 11244542 IC50 > 10000 nM T72267 CT8G0R 11338511 IC50 > 10000 nM T72267 CB26AX 11391631 IC50 > 10000 nM T72267 CFT60D 11475997 IC50 = 4610 nM T72267 C3L6FB 11748721 IC50 > 10000 nM T72267 C9C0DT 14898643 IC50 > 10000 nM T72267 C5RCD3 14898644 IC50 > 10000 nM T72267 C7Q8HG 14950683 IC50 > 10000 nM T72267 CG49IS 14950684 IC50 > 10000 nM T72267 CLK42M 14950685 IC50 > 10000 nM T72267 CD13NW 14950686 IC50 > 10000 nM T72267 C39MRN 15262805 IC50 > 10000 nM T72267 CZ7E3U 16067273 IC50 > 10000 nM T72267 CTL0C7 21858022 IC50 > 10000 nM T72267 CF2S3C 21858023 IC50 > 10000 nM T72267 CGN80J 23643046 IC50 = 9910 nM T72267 CN91XU 44806719 EC50 > 10000 nM T72267 C0BQ4U 49890666 IC50 > 10000 nM T72267 C0YH3T 70677671 IC50 > 10000 nM T72267 CR71AY 70677673 IC50 > 10000 nM T72267 CFMD45 70677677 IC50 > 10000 nM T72267 C2E1AD 70677804 IC50 > 10000 nM T72267 CCE2U9 70677807 IC50 > 10000 nM T72267 C74KDW 70677808 IC50 > 10000 nM T72267 CSGH58 70677953 IC50 > 10000 nM T72267 CCUW05 70677955 IC50 > 10000 nM T72267 CB4P6Y 70677956 IC50 > 10000 nM T72267 CV7Q3G 70677959 IC50 > 10000 nM T72267 C4Y1LE 70678097 IC50 = 8100 nM T72267 C3DX1U 70678098 IC50 > 10000 nM T72267 C71DQG 70678099 IC50 = 15900 nM T72267 CJ0P4V 70678100 IC50 > 10000 nM T72267 C82PMZ 70678101 IC50 = 12500 nM T72267 CTB19O 70678102 IC50 > 10000 nM T72267 C46QGZ 70678238 IC50 >= 10000 nM T72267 CBX9D4 70678239 IC50 > 10000 nM T72267 CS7FL4 70678240 IC50 >= 10000 nM T72267 CDJH76 71682490 IC50 > 10000 nM T72267 C48BSN 71682637 IC50 = 11300 nM T72267 C0O9HE 71682639 IC50 > 10000 nM T72267 CZE6R2 71682640 IC50 >= 10000 nM T72267 C2FBL9 71682641 IC50 > 10000 nM T72267 CTOL05 71682642 IC50 > 10000 nM T72267 CDX59H 71682795 IC50 >= 10000 nM T72267 C3S1OE 71682796 IC50 > 10000 nM T72267 CNM1Y8 71682797 IC50 > 10000 nM T72267 C0HS4I 71682799 IC50 = 10000 nM T72267 CK0Y3J 71682950 IC50 > 10000 nM T72267 CO4IL2 76317959 IC50 > 10000 nM T72267 C5GI9Z 76325292 IC50 = 13400 nM T72267 CQE10H 85468767 IC50 > 10000 nM T72267 CA0Y8G 85469571 IC50 = 279 nM T72267 CVY83X 90667465 IC50 = 6450 nM T72267 C85BUR 90667466 IC50 > 10000 nM T72267 C0FZU2 90667467 IC50 > 10000 nM T72267 C4MF8A 90667653 IC50 > 10000 nM T72267 CR2WI4 90667654 IC50 = 7220 nM T72267 C8N0LA 90667655 IC50 = 1650 nM T72267 CU23VX 90667656 IC50 = 2550 nM T72267 CR8I5E 90667657 IC50 = 6160 nM T72267 CI61LD 90667658 IC50 = 6350 nM T72267 C7P2EG 90667659 IC50 = 14300 nM T72267 CS5DZ4 90667660 IC50 = 10000 nM T72267 C31ZMH 90667661 IC50 > 10000 nM T72267 CT37YL 90667662 IC50 = 6480 nM T72267 CJ7V0Y 90667663 IC50 > 10000 nM T72267 C54BTS 90667664 IC50 > 10000 nM T72267 CJP21Z 90667665 IC50 > 10000 nM T72267 C9RM7U 90667666 IC50 > 10000 nM T72267 C1F0BP 145949413 EC50 > 10000 nM T72267 CBC13V 145949551 EC50 > 10000 nM T72267 CXRO20 145950071 IC50 = 2380 nM T72267 CY60SW 145951064 IC50 = 238 nM T72267 CCKN03 145951123 EC50 > 10000 nM T72267 CSG0W9 145951227 EC50 > 10000 nM T72267 C4LX7H 145951404 IC50 = 3590 nM T72267 C3G5TZ 145952824 IC50 = 1490 nM T72267 CS10GA 145953541 IC50 > 10000 nM T72267 CDI42H 145953879 IC50 = 650 nM T72267 C6QX5T 145954189 IC50 = 1150 nM T72267 CKO9B4 145954190 EC50 > 10000 nM T72267 COMQ03 145954409 EC50 > 10000 nM T72267 C03WAH 145954816 IC50 = 1730 nM T72267 CUE8Y2 145955444 EC50 > 10000 nM T72267 CX95DH 145955833 EC50 > 10000 nM T72267 CG16ZX 145956544 EC50 > 10000 nM T72267 CA30EJ 145956612 IC50 = 1710 nM T72267 CW3A0Y 145958034 IC50 = 13800 nM T72267 CIK3B7 145958405 IC50 = 10000 nM T72267 CC5B9Y 145958428 IC50 = 3250 nM T72267 C3IH1U 145958480 IC50 = 2290 nM T72267 COP8M1 145958551 EC50 > 10000 nM T72267 CEQ9W7 145958588 IC50 > 10000 nM T72267 C5K9TY 145959141 EC50 > 10000 nM T72267 C25WFH 145960085 EC50 > 10000 nM T72267 CQ3B6P 145960178 IC50 = 5000 nM T72267 C5T2WE 145971274 IC50 = 4780 nM T72267 C6XAW4 145971463 IC50 > 10000 nM T72267 C4G8WI 145974549 IC50 = 1140 nM T72267 D01RWS 16066912 IC50 > 10000 nM T72267 D01ZHW 5283389 EC50 = 20 nM T72267 D08MON 16067266 IC50 > 10000 nM T72267 D0D6OH 104895 EC50 = 5990 nM T85221 C8INU2 6861581 IC50 = 1500 nM T85221 CE9Y0L 6869187 IC50 = 1100 nM T85221 CQ9GJ2 9690663 IC50 = 240 nM T85221 CO1XF3 9690863 IC50 > 100000 nM T85221 CM15OG 9729606 IC50 > 100000 nM T85221 CG41FJ 9777510 IC50 = 100000 nM T85221 C42WPQ 9817849 IC50 = 10000 nM T85221 CVCO26 9818018 IC50 = 1500 nM T85221 C9XZT2 9864110 IC50 > 100000 nM T85221 CD6QX7 9882828 IC50 = 17000 nM T85221 CK19TA 9905084 IC50 = 330 nM T85221 C47SDT 9927509 IC50 = 220 nM T85221 CZG9D5 9951194 IC50 = 2000 nM T85221 C1DR5A 11724855 IC50 = 170 nM T85221 CE1B6K 44308616 IC50 = 3700 nM T85221 C7EZI0 44308842 IC50 > 100000 nM T85221 CO0AX1 44308851 IC50 > 50000 nM T85221 COT8H6 44308854 IC50 = 2400 nM T85221 CQA6N3 44308856 IC50 = 16000 nM T85221 C6E4VF 44308873 IC50 = 25000 nM T85221 CT1YG3 44308949 IC50 = 700 nM T85221 C32DRP 44308982 IC50 = 25000 nM T85221 C2U3XP 44591656 IC50 = 79000 nM T85221 C10LIG 135409477 IC50 = 2400 nM T34234 D03ZTE 10133 EC50 > 150000 nM T34234 D05BTM 6398761 EC50 = 0.855 nM T34234 D08SVH 5283734 EC50 = 7.05 nM T34234 D0G3SH 31401 EC50 > 150000 nM T34234 D0K5WS 5280795 EC50 = 0.21 nM T34234 D0OR2L 221493 EC50 > 150000 nM T34234 D0T2PL 5280453 EC50 = 0.01 nM T34234 D02PQB 222528 EC50 > 150000 nM T34234 D04SLF 9903 EC50 = 2140 nM T34234 CPBA32 92880 IC50 = 15100 nM T34234 CXQ5O3 115245 IC50 = 40100 nM T34234 CC4X3R 451489 IC50 = 23300 nM T34234 C2UP4X 888443 IC50 = 14200 nM T34234 CEP9X8 888651 IC50 = 28000 nM T34234 CT3S5C 2153736 IC50 = 13700 nM T34234 C1KO0D 2173330 IC50 = 21600 nM T34234 CL2EG5 2196926 IC50 = 10500 nM T34234 CMRS49 2201555 IC50 = 37600 nM T34234 C4U9OV 3133586 IC50 = 28900 nM T34234 C9XF0N 3262522 IC50 = 15300 nM T34234 CDZ6P1 3262523 IC50 = 14100 nM T34234 CQ4EJ2 3262524 IC50 = 22100 nM T34234 C0YJ6D 3422053 IC50 = 17200 nM T34234 C2ZC7Y 3456940 IC50 = 27700 nM T34234 C4IG6O 3590557 IC50 = 25100 nM T34234 CHT60N 3631309 IC50 = 9500 nM T34234 C4VOW1 3943163 IC50 = 3200 nM T34234 CYD04S 4109852 IC50 = 25000 nM T34234 CI7YP4 4124316 IC50 = 51500 nM T34234 CL8RJ0 4177080 IC50 > 75000 nM T34234 C3C8ZA 4386676 IC50 = 2000 nM T34234 C5G1ES 4613666 IC50 = 30300 nM T34234 C9G8HR 5283820 EC50 > 150000 nM T34234 C16ZSG 6439929 IC50 = 2000 nM T34234 CEM24L 7203539 EC50 = 1490 nM T34234 CMY18Z 9547273 EC50 = 870 nM T34234 C74HDM 9547693 IC50 = 6 nM T34234 CB53GZ 9806383 EC50 = 0.35 nM T34234 CS51DP 9844459 EC50 = 49 nM T34234 C5UVH8 9847095 EC50 = 0.5 nM T34234 CR8X2M 10174128 EC50 = 2.2 nM T34234 C89SWQ 10437131 IC50 = 700 nM T34234 C3TAS4 11341817 IC50 = 194 nM T34234 CULO82 11505040 IC50 = 2200 nM T34234 C94HOT 11531991 EC50 = 0.68 nM T34234 CRBK17 11584775 IC50 = 220 nM T34234 CLV13I 11606649 IC50 = 390 nM T34234 CB6C4Y 11611620 EC50 = 150 nM T34234 C0WX9D 11775402 IC50 = 6 nM T34234 C7YJM3 11957208 IC50 = 6800 nM T34234 C9CQF7 11993876 IC50 = 9.3 nM T34234 C87APF 11993877 IC50 = 8.6 nM T34234 C6PB7F 11993878 IC50 = 6 nM T34234 C80IKL 11993879 IC50 = 8.2 nM T34234 CO0QR3 11993880 IC50 = 8.6 nM T34234 CNHF07 11993881 IC50 = 6 nM T34234 CS9F1Q 11993998 IC50 = 10.25 nM T34234 C5NQ7X 11993999 IC50 = 6.8 nM T34234 C5JX6Z 11994000 IC50 = 6.2 nM T34234 CEP41H 11994001 IC50 = 6.7 nM T34234 CQFE46 11994002 IC50 = 8.4 nM T34234 CKN0V1 11994003 IC50 = 6.3 nM T34234 CU98FC 11994125 IC50 = 6.7 nM T34234 C2J9RO 11994126 IC50 = 8.8 nM T34234 CM9CO4 11994127 IC50 = 10.5 nM T34234 C3CVO8 11994128 IC50 = 9.3 nM T34234 CJ3F9E 11994129 IC50 = 6.2 nM T34234 C2CB4F 11994261 IC50 = 6.7 nM T34234 CNGM18 11994262 IC50 = 8.4 nM T34234 CTOQ18 11994263 IC50 = 6.3 nM T34234 C0S2GI 11994264 IC50 = 6.3 nM T34234 CDRE79 11994265 IC50 = 8.8 nM T34234 CY67TB 11994398 IC50 = 11 nM T34234 CA68ZP 11994399 IC50 = 9.3 nM T34234 C49NHG 11994400 IC50 = 8.1 nM T34234 CCTZ26 11994401 IC50 = 6.1 nM T34234 CO21GE 11994402 IC50 = 8.4 nM T34234 C8K2HD 11994522 IC50 = 8.4 nM T34234 C2T7YU 11994523 IC50 = 6.3 nM T34234 CO3JG7 11994524 IC50 = 6.7 nM T34234 CKC9D3 11994525 IC50 = 8.8 nM T34234 CYTK52 11994526 IC50 = 9.3 nM T34234 C1KPA6 11994644 IC50 = 9.3 nM T34234 CXRG61 11994645 IC50 = 6.2 nM T34234 CYS81N 11994646 IC50 = 6.7 nM T34234 CP16WI 11994647 IC50 = 8.4 nM T34234 C9LZ3E 11994648 IC50 = 6.3 nM T34234 CKJ08L 11994765 IC50 = 6.3 nM T34234 CW6IM2 11994766 IC50 = 8.8 nM T34234 CV6B3W 11994767 IC50 = 10.55 nM T34234 C95WCO 11994768 IC50 = 9.3 nM T34234 C65SRY 11994897 IC50 = 10.2 nM T34234 CKZM82 11994898 IC50 = 8.2 nM T34234 CHG51I 11995133 IC50 = 6.1 nM T34234 C4GD3Y 11995134 IC50 = 8.4 nM T34234 C8JT3Y 11995135 IC50 = 6.3 nM T34234 C9SRM8 11995234 IC50 = 6.3 nM T34234 CXSU20 11995235 IC50 = 8.8 nM T34234 CNI1P5 11995236 IC50 = 9.3 nM T34234 C2QIA9 11995237 IC50 = 6.8 nM T34234 C0U8OG 11995238 IC50 = 6.1 nM T34234 CSJ5K9 11995239 IC50 = 8.4 nM T34234 CF0XA5 11995338 IC50 = 6.3 nM T34234 CSFD67 11995339 IC50 = 6.7 nM T34234 C4T0OQ 11995340 IC50 = 8.8 nM T34234 C2HG0T 11995341 IC50 = 9.3 nM T34234 C0QXA2 11995435 IC50 = 6.2 nM T34234 CG0XY4 11995436 IC50 = 6.7 nM T34234 CFR94W 11995437 IC50 = 6.3 nM T34234 CN5L9F 11995438 IC50 = 6.3 nM T34234 CZY5U4 11995439 IC50 = 8.8 nM T34234 CD6HK3 11995440 IC50 = 11 nM T34234 C2E7CO 11995537 IC50 = 8.6 nM T34234 CJY2O4 11995538 IC50 = 8.1 nM T34234 CG1ZL4 11995539 IC50 = 6.1 nM T34234 C4MKF0 11995540 IC50 = 8.4 nM T34234 C1Q6LZ 11995541 IC50 = 6.3 nM T34234 C0ZUY1 11995542 IC50 = 6.7 nM T34234 CW69HF 11995632 IC50 = 6 nM T34234 C5ATF8 11995633 IC50 = 8.2 nM T34234 C3H2DV 11995634 IC50 = 9.5 nM T34234 C54KZE 11995635 IC50 = 8.6 nM T34234 C0DZY1 11995636 IC50 = 6 nM T34234 C2T6YV 11995637 IC50 = 8.2 nM T34234 C39IED 11995638 IC50 = 8.8 nM T34234 CY3KS1 11995639 IC50 = 9.3 nM T34234 C96KXP 15521394 EC50 = 40 nM T34234 C6O3IY 20222540 IC50 = 30200 nM T34234 C6VKG3 20647489 EC50 = 90 nM T34234 C89NTR 20876820 IC50 = 10500 nM T34234 CF3L9A 21771350 IC50 = 1200 nM T34234 CI9M7X 23605495 IC50 = 5300 nM T34234 CHS28Q 23605496 IC50 = 2600 nM T34234 C3W8DR 23605507 IC50 = 1600 nM T34234 CXK39R 23605513 IC50 = 6200 nM T34234 CHY64Z 23656120 IC50 = 85 nM T34234 CD59KP 23656626 IC50 = 198 nM T34234 CCWB72 23656628 IC50 = 63 nM T34234 COEP93 23656791 IC50 = 47 nM T34234 CTE1N2 24748569 EC50 > 10000 nM T34234 C0PD6R 24883478 EC50 = 0.02 nM T34234 C4BX5H 24883479 EC50 = 1 nM T34234 C6MZ7I 24883480 EC50 = 24 nM T34234 C97QRS 24936209 EC50 = 0.0396 nM T34234 C6BDX3 25207860 IC50 = 185 nM T34234 C1HO8K 25210169 IC50 = 107 nM T34234 CE3Y2C 42624365 EC50 = 0.69 nM T34234 C9F2OB 44301422 EC50 = 0.18 nM T34234 C79WPU 44409491 IC50 > 2000 nM T34234 CF7HX4 44409495 IC50 > 1000 nM T34234 C0ZN4Y 44409509 IC50 = 2200 nM T34234 C9MC1H 44409561 IC50 = 390 nM T34234 C67PDU 44409588 IC50 = 700 nM T34234 C7BSE3 44409634 IC50 = 207 nM T34234 CY4L1H 44409642 IC50 = 660 nM T34234 C3HN9U 44417670 IC50 = 6 nM T34234 C9IAR5 44417671 IC50 = 11 nM T34234 CM61HP 44417674 IC50 = 7.7 nM T34234 CEWC01 44417679 IC50 = 7.7 nM T34234 C9XG0S 44417690 IC50 = 9.2 nM T34234 C1O8DM 44418743 IC50 = 30 nM T34234 CF7W3S 44420574 EC50 = 0.003 nM T34234 C4E8FB 44420575 EC50 = 0.002 nM T34234 CU96LK 44420576 EC50 = 0.2 nM T34234 CCPR87 44423318 EC50 = 0.5 nM T34234 CVA9R4 44423319 EC50 = 0.07 nM T34234 CZM0B4 44436706 IC50 = 300 nM T34234 CUK1N9 44451424 EC50 = 10 nM T34234 C6P4QJ 44451449 EC50 = 6 nM T34234 CZM79P 44451450 EC50 = 1 nM T34234 CZ1Y7T 44455867 EC50 = 15.6 nM T34234 C8I4CF 44455886 EC50 = 4.68 nM T34234 CBV4A3 44455888 EC50 = 1.66 nM T34234 CR5SI0 44476535 EC50 > 10000 nM T34234 CF06LW 44578181 IC50 = 300 nM T34234 C7WEF5 44578182 IC50 > 3000 nM T34234 CY06EB 44578183 IC50 > 3000 nM T34234 C60NEH 44578184 IC50 > 3000 nM T34234 CJ6ES8 44578185 IC50 = 860 nM T34234 CHUG86 44578189 IC50 = 780 nM T34234 C45KPD 44578206 IC50 = 90 nM T34234 CN83PX 44578207 IC50 = 180 nM T34234 CS4M1I 44578208 IC50 = 540 nM T34234 C35HAR 46261199 IC50 = 20500 nM T34234 CDV4P2 46499637 IC50 = 6000 nM T34234 CCUR46 46499640 IC50 = 5700 nM T34234 C12ZFM 46500390 IC50 = 8600 nM T34234 C40WCI 46500406 IC50 = 3900 nM T34234 CZPL02 46866395 IC50 = 13000 nM T34234 C7Q6ZD 46866396 IC50 = 28000 nM T34234 CL6SY4 46866497 IC50 = 17000 nM T34234 CDHA57 46880834 IC50 = 30000 nM T34234 C5LY0E 46880871 IC50 > 30000 nM T34234 C9P8TB 46880920 IC50 > 30000 nM T34234 CU7L5W 46906597 IC50 = 280 nM T34234 CG46KJ 46906641 IC50 = 196 nM T34234 C4V7PG 46907052 IC50 = 87 nM T34234 CMQ3R0 46907054 IC50 = 248 nM T34234 C05KTS 46907124 IC50 = 524 nM T34234 C2PC1Z 46907160 IC50 = 36 nM T34234 C72BEW 46907196 IC50 = 213 nM T34234 C4V3ZK 46907197 IC50 = 321 nM T34234 C6TRS7 46907198 IC50 = 14 nM T34234 C0K4DL 46907280 IC50 = 29 nM T34234 C3NE0Q 46907281 IC50 = 15 nM T34234 CJ3FM4 46925833 EC50 = 1950 nM T34234 CUD91T 49862248 EC50 > 10000 nM T34234 CE82QV 50899366 EC50 = 3600 nM T34234 CLMP79 52940658 EC50 > 30000 nM T34234 C2XB9F 52940978 EC50 = 21000 nM T34234 C6GH0Z 52943083 EC50 > 30000 nM T34234 CTP2Z0 52943284 EC50 = 7100 nM T34234 CX0J1E 52944485 EC50 = 22000 nM T34234 COEG38 52944493 EC50 > 30000 nM T34234 C6T0PY 52944539 EC50 > 30000 nM T34234 CX5PG4 52945275 EC50 > 30000 nM T34234 CX2BF4 52945709 EC50 > 30000 nM T34234 CT28DY 52945795 EC50 = 23000 nM T34234 CH87CZ 52946714 EC50 > 30000 nM T34234 CCPU06 52946931 EC50 = 11000 nM T34234 CQAF42 52949161 EC50 > 30000 nM T34234 C5TYU7 56603803 EC50 = 0.06 nM T34234 CS7PI3 56666231 EC50 = 19.4 nM T34234 CB9UG1 56666232 EC50 = 1.25 nM T34234 CJD8G2 56666233 EC50 = 1.29 nM T34234 C6J9FV 56669637 EC50 = 0.92 nM T34234 CIS46N 56679790 EC50 = 1.11 nM T34234 C8A3BM 57522254 IC50 = 0.029 nM T34234 C1HO3L 57522255 IC50 = 0.38 nM T34234 C7M2PI 57522256 IC50 = 0.41 nM T34234 C64MWB 57824615 IC50 = 1.13 nM T34234 CWPJ42 59263691 EC50 = 1.7 nM T34234 CF4GR9 59263692 EC50 = 5 nM T34234 C28PFQ 66550229 IC50 = 25400 nM T34234 C1DC7M 69734881 EC50 = 850 nM T34234 C3Z2WN 70682577 IC50 = 14600 nM T34234 C7TAC0 70682578 IC50 = 13500 nM T34234 CKQ63R 70682579 IC50 = 13100 nM T34234 CZK0I2 70682580 IC50 > 70000 nM T34234 C67YPN 70684663 IC50 = 5800 nM T34234 CFVA95 70684664 IC50 = 8700 nM T34234 CA3XQ5 70684665 IC50 = 8600 nM T34234 CO51WT 70686813 IC50 = 24000 nM T34234 CR03AT 70688889 IC50 = 12200 nM T34234 CA05SM 70688890 IC50 = 8500 nM T34234 CKLD97 70688891 IC50 > 70000 nM T34234 CZBU30 70690978 IC50 = 31700 nM T34234 CM0TN7 70690979 IC50 = 20100 nM T34234 CFOB26 70690980 IC50 = 15000 nM T34234 CQ3K4Z 70690981 IC50 = 17700 nM T34234 CBX32O 70693111 IC50 = 4400 nM T34234 C21TPU 70695167 IC50 = 21600 nM T34234 CK82MV 70697216 IC50 = 12100 nM T34234 C3DIT2 71451627 IC50 = 3 nM T34234 C4D0OX 71451767 EC50 = 5.74 nM T34234 C86DRX 71457095 EC50 = 9.04 nM T34234 CL1SJ3 71460762 EC50 = 8.19 nM T34234 C4V8HD 71484079 EC50 = 0.07 nM T34234 CQ8M2Z 71524564 IC50 = 24000 nM T34234 C8K5RD 71524565 IC50 = 14000 nM T34234 CN4RX0 71524566 IC50 > 30000 nM T34234 C5PK9J 71524567 IC50 = 20000 nM T34234 C9L2WU 71524569 IC50 > 30000 nM T34234 CC1U5Z 71524615 IC50 > 30000 nM T34234 CX8H1A 71524616 IC50 > 30000 nM T34234 CPVM05 71524617 IC50 > 30000 nM T34234 CW3HC1 71524619 IC50 > 30000 nM T34234 CJ6R3Z 71524665 IC50 = 25000 nM T34234 C5CRN4 71524666 IC50 > 30000 nM T34234 C5LM6N 71525260 IC50 > 30000 nM T34234 C4ROL7 71525261 IC50 > 30000 nM T34234 C0J6VG 71525262 IC50 > 30000 nM T34234 CX06WI 71525263 IC50 > 30000 nM T34234 CD4JX5 71525264 IC50 = 30000 nM T34234 CDX57G 71563370 EC50 = 1.5 nM T34234 CYB0D9 71563371 EC50 = 0.8 nM T34234 CGHD73 71570928 IC50 > 60000 nM T34234 C49SBQ 71571065 IC50 > 60000 nM T34234 CE06XT 71571066 IC50 > 60000 nM T34234 CR92GT 71571067 IC50 > 60000 nM T34234 CTUC72 71571068 IC50 > 60000 nM T34234 C7UHM3 71571069 IC50 = 7000 nM T34234 C1P5HY 71571070 IC50 > 60000 nM T34234 C4CNP2 71571213 IC50 > 60000 nM T34234 CAV18D 71571215 IC50 > 60000 nM T34234 C97ISQ 71571216 IC50 > 60000 nM T34234 CC08YH 71583283 EC50 = 40 nM T34234 C5ZT9O 71716541 IC50 > 60000 nM T34234 C1TN8C 71716542 IC50 > 60000 nM T34234 CPJ4T2 71716543 IC50 > 60000 nM T34234 CP9B4C 71716544 IC50 > 60000 nM T34234 C4OE3H 71716545 IC50 > 60000 nM T34234 CIJ84X 71716546 IC50 > 60000 nM T34234 C4XL7Z 71716547 IC50 > 60000 nM T34234 C7BMG8 71716548 IC50 > 60000 nM T34234 C8O2NJ 71716549 IC50 > 60000 nM T34234 CA1Q0X 71716550 IC50 > 60000 nM T34234 CM6ZN5 71716551 IC50 > 60000 nM T34234 CX6RH7 71716552 IC50 > 60000 nM T34234 CTI7H2 71716553 IC50 > 60000 nM T34234 C8YEZ6 71716554 IC50 > 60000 nM T34234 CT3D1M 71717145 IC50 > 60000 nM T34234 CSHP85 71717146 IC50 > 60000 nM T34234 C5K3QG 71717147 IC50 = 66000 nM T34234 C6B5DO 71717148 IC50 > 60000 nM T34234 CK0ZQ9 71717149 IC50 > 60000 nM T34234 C96GSC 71717150 IC50 > 60000 nM T34234 C36SFW 71717155 IC50 > 60000 nM T34234 CLR58A 71717156 IC50 > 60000 nM T34234 CN4A9V 71717771 IC50 > 60000 nM T34234 CPLW58 71717772 IC50 > 60000 nM T34234 CIL03B 71717773 IC50 > 60000 nM T34234 C63QLG 71717774 IC50 > 60000 nM T34234 CV0I1H 71717775 IC50 = 38000 nM T34234 CUN4O0 71717776 IC50 > 60000 nM T34234 CSO2X5 71717777 IC50 > 60000 nM T34234 C52BZC 71717778 IC50 > 60000 nM T34234 CIE8V5 71717779 IC50 > 60000 nM T34234 C46ICD 71717780 IC50 > 60000 nM T34234 CPH02C 71718378 IC50 = 50000 nM T34234 COX71E 71718379 IC50 > 60000 nM T34234 CC94QZ 71718380 IC50 = 51000 nM T34234 CG2TH9 71718381 IC50 > 60000 nM T34234 C6G4BT 71718382 IC50 = 40000 nM T34234 CQ8AI1 71718383 IC50 > 60000 nM T34234 C4KOT9 71718386 IC50 > 60000 nM T34234 CH2TV1 71718387 IC50 > 60000 nM T34234 CXO1S7 71718388 IC50 > 60000 nM T34234 CI6AN0 71718985 IC50 > 60000 nM T34234 C5U7IR 71718986 IC50 > 60000 nM T34234 C0CJ8S 71718987 IC50 > 60000 nM T34234 C4KAZ7 71718988 IC50 = 65000 nM T34234 CIN3V1 71718992 IC50 > 60000 nM T34234 CZ3WG5 71718993 IC50 > 60000 nM T34234 CE6X2K 71718994 IC50 > 60000 nM T34234 C1IH2Q 71718995 IC50 > 60000 nM T34234 CN1RW4 71718996 IC50 > 60000 nM T34234 CKA36P 71718997 IC50 > 60000 nM T34234 C8LWP5 71719585 IC50 > 60000 nM T34234 CQ6BL0 71719586 IC50 > 60000 nM T34234 CFO1J2 71719587 IC50 > 60000 nM T34234 CT0DH9 71719588 IC50 > 60000 nM T34234 C3BT7V 71719589 IC50 > 60000 nM T34234 CBY36L 71719590 IC50 > 60000 nM T34234 C5SPB2 71719591 IC50 > 60000 nM T34234 CYNI30 71719592 IC50 > 60000 nM T34234 CJ5O6Q 71719593 IC50 > 60000 nM T34234 C7EKV1 71719594 IC50 > 60000 nM T34234 CB7O4D 71719597 IC50 > 60000 nM T34234 CD98PS 71719598 IC50 > 60000 nM T34234 CQ7U4O 71719599 IC50 > 60000 nM T34234 CXDE81 71719600 IC50 > 60000 nM T34234 CDM58X 71719601 IC50 > 60000 nM T34234 CCV8I1 71719602 IC50 > 60000 nM T34234 CH1EB5 71719603 IC50 > 60000 nM T34234 CX46KH 71719604 IC50 > 60000 nM T34234 C7KER0 71720182 IC50 = 37000 nM T34234 C0DYJ3 71720183 IC50 = 44000 nM T34234 CY4J2C 71720184 IC50 > 60000 nM T34234 C4Z0VS 71720185 IC50 > 60000 nM T34234 C5H0WP 71720186 IC50 > 60000 nM T34234 C9B4SP 71720187 IC50 > 60000 nM T34234 CHFZ51 71720188 IC50 > 60000 nM T34234 C2FM0U 71720189 IC50 > 60000 nM T34234 CUG52N 71720190 IC50 > 60000 nM T34234 CV1US9 71720192 IC50 > 60000 nM T34234 C7X8QB 71720193 IC50 > 60000 nM T34234 CB56IU 71720826 IC50 = 55000 nM T34234 CS5R7G 71720827 IC50 > 60000 nM T34234 CTF8D3 71720828 IC50 > 60000 nM T34234 CZ71PL 71720830 IC50 > 60000 nM T34234 C0Y9CT 71720831 IC50 > 60000 nM T34234 C1XW8N 71725364 IC50 = 600000 nM T34234 CRN3M1 71725365 IC50 = 520000 nM T34234 CJ6XZ7 71725438 IC50 = 220000 nM T34234 C5FX2V 71725439 IC50 = 3200 nM T34234 C7SY0M 71725531 IC50 = 610000 nM T34234 CXQ7H4 71725532 IC50 = 430000 nM T34234 C04GPB 71725533 IC50 = 610000 nM T34234 C1M5JH 71764798 EC50 = 0.01 nM T34234 CQ96JL 71764799 EC50 = 0.29 nM T34234 CV3G1O 71764800 EC50 = 0.15 nM T34234 C9R5BI 71764801 EC50 = 0.044 nM T34234 C4RWM0 71765011 EC50 = 0.21 nM T34234 CC93OP 71765012 EC50 = 0.68 nM T34234 CFTY60 73334809 IC50 = 590 nM T34234 C05FCR 73346485 EC50 = 110 nM T34234 C3NX7U 73346488 EC50 = 410 nM T34234 C63FLS 73346489 EC50 = 790 nM T34234 C0HSC8 73346520 Ki = 2840 nM T34234 C8SD9P 73346521 Ki = 24440 nM T34234 CGZ6Y8 73346522 Ki = 4130 nM T34234 CGEV82 73347982 EC50 = 1.06 nM T34234 C43IPQ 73348006 Ki = 3660 nM T34234 CNPO14 73349524 EC50 = 1600 nM T34234 CV24HD 73349525 EC50 = 1830 nM T34234 CA49EI 73349527 EC50 = 23 nM T34234 C36ZVJ 73351080 EC50 = 5640 nM T34234 CS9C0W 73351108 Ki = 17080 nM T34234 C3V4CZ 73352548 EC50 = 4950 nM T34234 CT35PK 73352550 EC50 = 33220 nM T34234 C14DJK 73352551 EC50 = 150 nM T34234 C27JUH 73352576 Ki = 2280 nM T34234 CVP03Z 73352577 Ki = 28250 nM T34234 CDAB86 73354065 Ki = 1030 nM T34234 CK3Z8U 73354066 Ki = 1600 nM T34234 C92DXZ 73354067 Ki = 13680 nM T34234 C1V4KY 73355572 EC50 = 4.07 nM T34234 COZ64C 73355573 EC50 = 570 nM T34234 CVT98N 73355574 EC50 = 200 nM T34234 CCI18Y 73355591 Ki = 3070 nM T34234 CRX8A0 73355592 Ki = 4660 nM T34234 C4Z3ER 73357083 EC50 < 0.1 nM T34234 COMV71 73357115 EC50 = 2630 nM T34234 CVJ6D7 74331693 IC50 = 0.29 nM T34234 C35PDL 74331694 IC50 = 1.79 nM T34234 CF3L7E 76310292 IC50 = 5800 nM T34234 C92XAR 76310293 IC50 = 15800 nM T34234 C70UYQ 76310294 IC50 = 8500 nM T34234 C70LFD 76310295 IC50 = 590 nM T34234 C27TWJ 76313972 IC50 = 9300 nM T34234 CY7SE1 76317515 IC50 = 3200 nM T34234 CG3T1E 76317516 IC50 = 3800 nM T34234 CDY64J 76321238 IC50 = 4400 nM T34234 CY4SH5 76321239 IC50 = 7200 nM T34234 C0QC8N 76321240 IC50 = 9100 nM T34234 CSE0H6 76321241 IC50 = 32300 nM T34234 CANR79 76324858 IC50 = 5000 nM T34234 C98EGF 76324859 IC50 = 3400 nM T34234 CXU31F 76324861 IC50 > 25000 nM T34234 CND2E7 76328416 IC50 = 5800 nM T34234 C5KYG3 76328417 IC50 = 14200 nM T34234 CE9W6N 76328418 IC50 = 6700 nM T34234 C5RWN2 76332098 IC50 = 6100 nM T34234 CES0Z2 76335714 IC50 = 3000 nM T34234 CFY25B 76335715 IC50 = 22800 nM T34234 C0BF2I 76335716 IC50 = 5200 nM T34234 C9CL2H 76335717 IC50 = 7300 nM T34234 CK29WF 76335718 IC50 = 66800 nM T34234 C5IOG1 76335719 IC50 = 12200 nM T34234 CJG1Y3 90656368 IC50 = 0.26 nM T34234 CIS18W 90656369 IC50 = 2.87 nM T34234 CXCJ07 90656370 IC50 = 0.12 nM T34234 C7DT3J 90656371 IC50 = 1.55 nM T34234 C3QI2P 90656372 IC50 = 0.89 nM T34234 CQDO74 90656373 IC50 = 7.16 nM T34234 C8J0OB 90656374 IC50 = 2.39 nM T34234 CQ21MO 90656375 IC50 = 1.55 nM T34234 C0DOG2 90656755 EC50 = 4 nM T34234 C6OMI1 91799374 IC50 = 4.5 nM T34234 C0DQ4K 92045001 IC50 = 0.21 nM T34234 CO3Z1B 100945784 IC50 = 2860 nM T34234 CY6W8K 101585746 EC50 > 10000 nM T34234 CB2UX7 101627374 EC50 = 12300 nM T34234 C6KXC7 112499899 IC50 = 0.09 nM T34234 CU3K9N 118101130 EC50 = 10 nM T34234 C3W7TH 118101135 EC50 = 29 nM T34234 CZ5O8N 118101158 EC50 = 8.6 nM T34234 C92YLG 118101159 EC50 = 9 nM T34234 C6R0HK 118719211 IC50 = 50 nM T34234 CJ5PE8 118727102 IC50 = 500000 nM T34234 CE24KA 118727103 IC50 = 67000 nM T34234 C2HVJ4 118727104 IC50 = 20000 nM T34234 C6TBD2 121345502 EC50 > 20000 nM T34234 CQ0WY5 122192534 EC50 = 64.9 nM T34234 CR2KO4 122192535 EC50 = 207.9 nM T34234 CY98DO 122195385 EC50 = 1500 nM T34234 C7QMK1 122195510 EC50 = 1200 nM T34234 C8O4YE 122195511 EC50 > 3000 nM T34234 C26OAH 122227448 EC50 = 4100 nM T34234 CM7N8H 122227450 EC50 = 3700 nM T34234 C25NTW 127037933 EC50 = 77 nM T34234 C3HRP4 127037934 EC50 = 96 nM T34234 CJXE94 127037939 EC50 = 22 nM T34234 CEF3I0 127037940 EC50 = 2200 nM T34234 C0EU8K 127037967 EC50 = 20 nM T34234 CFMC03 127038301 EC50 = 130 nM T34234 C0GKU5 127038302 EC50 = 240 nM T34234 CN8BJ1 127038303 EC50 = 1900 nM T34234 CK7RX6 127038952 EC50 = 14 nM T34234 CRG68P 127038953 EC50 = 37 nM T34234 CZ19RJ 127039266 EC50 = 66 nM T34234 CE0S6J 127039267 EC50 = 150 nM T34234 CAMQ12 127039268 EC50 = 18 nM T34234 C8WPF9 127039600 EC50 = 130 nM T34234 C09NQX 127039601 EC50 = 10 nM T34234 CKV5J9 127039602 EC50 = 1960 nM T34234 CL0MV7 127039603 EC50 = 3950 nM T34234 CB54NK 127039604 EC50 = 6400 nM T34234 CHRC85 127039928 EC50 = 97 nM T34234 C2WJE6 127039937 EC50 = 200 nM T34234 CM3L5W 127039938 EC50 = 1030 nM T34234 C1A8ET 127039939 EC50 = 380 nM T34234 C7IVS4 127039940 EC50 = 10 nM T34234 C15ABZ 127040282 EC50 = 1390 nM T34234 CCHE80 127040283 EC50 = 2.3 nM T34234 CGJ90L 127040289 EC50 = 740 nM T34234 C3UWC4 127040290 EC50 > 50000 nM T34234 C2BA8F 127040291 EC50 > 50000 nM T34234 CR3DO4 127040292 EC50 > 50000 nM T34234 CHVO14 127040293 EC50 = 45600 nM T34234 CF6IC7 127041001 EC50 = 120 nM T34234 CO43DZ 127041002 EC50 = 9800 nM T34234 CSB51R 127041262 EC50 = 2320 nM T34234 C6JA8S 127041263 EC50 > 50000 nM T34234 CB5FD3 127041264 EC50 > 50000 nM T34234 CMHL57 127041265 EC50 = 630 nM T34234 CG9WN5 127041266 EC50 > 50000 nM T34234 CK3OT1 127041314 EC50 = 21600 nM T34234 CNO6D1 127041315 EC50 = 18500 nM T34234 C1W9UN 127041316 EC50 = 870 nM T34234 C6GR0N 127041319 EC50 = 210 nM T34234 CW9Q8N 127041320 EC50 = 28800 nM T34234 C0B1RJ 127041321 EC50 > 50000 nM T34234 CP9FY2 127041322 EC50 = 26 nM T34234 CYE4O1 127041323 EC50 = 210 nM T34234 CZBV93 127041324 EC50 = 6.54 nM T34234 C5GK3O 127041574 EC50 = 5100 nM T34234 C3N1VE 127041575 EC50 > 50000 nM T34234 C3R0NX 127041875 EC50 = 9500 nM T34234 CA8K6U 127041876 EC50 > 50000 nM T34234 CP1Y6U 127041877 EC50 > 50000 nM T34234 C0RBL2 127042154 EC50 = 240 nM T34234 C2C3UD 127042862 EC50 = 590 nM T34234 CBP2R4 127042863 EC50 > 50000 nM T34234 CP53QY 127042864 EC50 = 91 nM T34234 CAOD50 127042890 EC50 = 7 nM T34234 CWD9G8 127042891 EC50 = 30 nM T34234 C5CV4Q 127049261 EC50 = 484 nM T34234 C3KA8U 127049582 EC50 = 30.64 nM T34234 CI3X9L 127049803 EC50 = 510 nM T34234 C2O5LX 127049804 EC50 > 3000 nM T34234 CHEJ56 127051742 EC50 = 174.8 nM T34234 CP6WD0 134158367 IC50 = 20 nM T34234 CN1BD8 134158369 IC50 = 84 nM T34234 CQ9GJ7 134693734 EC50 = 0.03 nM T34234 CKNY80 134693735 IC50 = 1.75 nM T34234 CA95MF 134693767 IC50 = 2.3 nM T34234 CBRQ76 137348831 IC50 = 1.1 nM T34234 CU76EY 137348836 IC50 = 1.8 nM T34234 CAU30I 137633097 EC50 > 50 nM T34234 CE9N4Q 137634840 EC50 = 52.74 nM T34234 CFX94S 137635673 EC50 = 9.36 nM T34234 CLR93H 137636145 EC50 = 68.91 nM T34234 C8K9FX 137636662 IC50 = 23 nM T34234 C3LT8R 137636693 EC50 = 21 nM T34234 C1V8EA 137637845 IC50 = 520 nM T34234 CR6BY2 137637855 EC50 = 12.68 nM T34234 CNGQ52 137638580 EC50 > 10000 nM T34234 CBD5A9 137639585 EC50 = 54.33 nM T34234 CZ93KT 137640144 EC50 = 293.44 nM T34234 CE1P6T 137640606 EC50 = 1630 nM T34234 CGV4K7 137641102 IC50 = 400 nM T34234 CE4Y0H 137641111 EC50 = 450 nM T34234 C1TY7F 137641302 EC50 = 5 nM T34234 C86GCD 137641457 EC50 = 17.67 nM T34234 CN1E8T 137641740 EC50 = 82 nM T34234 CSQ32Y 137643553 EC50 = 96 nM T34234 C38ARI 137643845 EC50 > 10000 nM T34234 CANM93 137644540 EC50 = 10.12 nM T34234 C8PC1W 137644909 IC50 = 36 nM T34234 C6LCY1 137645203 EC50 = 2494 nM T34234 CJO6T0 137645523 EC50 > 50 nM T34234 CZX08W 137645781 EC50 = 12.56 nM T34234 CBU7Q4 137646538 EC50 > 50 nM T34234 CB2JA8 137647571 EC50 = 68.32 nM T34234 C41FLC 137648080 EC50 = 287.65 nM T34234 C6DQ1W 137648198 EC50 = 520 nM T34234 CBQ47Z 137648641 EC50 = 156 nM T34234 CE3B6P 137648901 EC50 = 1080 nM T34234 C7O9GT 137649139 IC50 = 17 nM T34234 CY91PT 137649490 EC50 = 19.29 nM T34234 CNH5M0 137649849 EC50 = 2653 nM T34234 C0GHN9 137650140 EC50 > 50 nM T34234 C6YXT0 137650434 EC50 > 10000 nM T34234 CLQ27P 137650892 EC50 = 11.36 nM T34234 CH15QY 137651328 EC50 = 26 nM T34234 C5A4IZ 137654603 IC50 = 102 nM T34234 C7HXA1 137654862 EC50 = 860 nM T34234 C1CXF4 137654924 EC50 = 142.17 nM T34234 C8VI7Q 137655186 EC50 = 5900 nM T34234 C6YWK2 137655366 EC50 > 50 nM T34234 CAJS52 137656336 EC50 > 10000 nM T34234 C1MU5A 137657397 EC50 = 6.98 nM T34234 CFDX92 137658518 EC50 = 8.5 nM T34234 CF2Z1C 137658922 EC50 = 238 nM T34234 C79WOV 137660092 EC50 = 66 nM T34234 CUAL38 137660277 EC50 > 50 nM T34234 C2AV8G 137660319 EC50 = 7.33 nM T34234 CQF32V 137660583 EC50 = 6033 nM T34234 CP6UI1 137660847 EC50 = 89 nM T34234 C20YAU 137661050 EC50 > 10000 nM T34234 CP5E4N 137661176 EC50 > 50 nM T34234 CF92KT 137661566 IC50 = 123.43 nM T34234 CJDA28 137662182 EC50 = 2.3 nM T34234 C1XM9S 145954006 IC50 = 1.9 nM T34234 C4BGJ9 145963928 IC50 = 5560 nM T34234 CCF02H 145964530 IC50 = 3820 nM T34234 C56SHA 145964597 IC50 = 5670 nM T34234 COLC12 145964669 IC50 = 10100 nM T34234 C2SKC3 145964785 IC50 = 6750 nM T34234 C5H8EZ 145965425 IC50 = 660 nM T34234 CC3X5W 145965684 IC50 > 80000 nM T34234 CB5Z9S 145965895 IC50 > 80000 nM T34234 C6BSE0 145965984 IC50 = 3350 nM T34234 CHP5B6 145970080 IC50 = 2880 nM T34234 CK1MR7 145972041 IC50 > 100000 nM T34234 CULX72 145973067 IC50 = 3250 nM T34234 CX06DP 145974139 IC50 = 3600 nM T34234 CEZA82 145974732 IC50 = 33140 nM T34234 CG1XZ6 145975539 IC50 > 80000 nM T34234 CH71OQ 145975878 IC50 > 33000 nM T34234 C5IXY0 145976191 IC50 = 4850 nM T34234 CUB0I8 145977098 IC50 > 80000 nM T34234 C98CHS 145977976 IC50 = 2500 nM T34234 C9B0GO 145978087 IC50 > 80000 nM T34234 CY5P0L 145988241 IC50 = 125.4 nM T34234 CCT5L1 145989687 IC50 = 89.1 nM T34234 CTX6P3 155511229 EC50 = 17.2 nM T34234 C8G6DQ 155512501 EC50 = 41.7 nM T34234 CN14MF 155520127 EC50 = 163 nM T34234 C75MXJ 155520322 EC50 = 76.9 nM T34234 COP7X8 155539171 IC50 > 10000 nM T34234 CSC42R 155548806 EC50 = 18 nM T34234 CX82TL 155557531 EC50 = 76.5 nM T34234 CL5P6C 155566184 EC50 = 9.26 nM T34234 D02CWP 439763 IC50 = 14500 nM T34234 D07AHG 15521397 EC50 = 40 nM T34234 D0D6XV 9547692 IC50 = 6.3 nM T34234 D0X0AM 9936230 EC50 = 0.4 nM T34234 D0X3DK 16094778 IC50 = 50 nM T34234 D0XZ2P 16094779 IC50 = 19.5 nM T73184 D00TLN 2913 Ki = 15000 nM T73184 C2JVZ1 4822 IC50 = 4300 nM T73184 CLV14X 95734 IC50 = 94600 nM T73184 CM0UP1 168897 IC50 = 59100 nM T73184 C98XBT 230362 IC50 > 100000 nM T73184 CWA90K 524039 IC50 > 100000 nM T73184 CEZ8D6 822743 IC50 = 30040 nM T73184 CQEF34 1002773 IC50 > 100000 nM T73184 C3FW7G 1740582 IC50 = 189700 nM T73184 CZV68S 2233086 IC50 = 4880 nM T73184 C4DJ3F 2258873 IC50 = 4590 nM T73184 CL3XN1 5237229 IC50 = 61750 nM T73184 CR0LH9 10039173 IC50 = 16300 nM T73184 CW39ZL 13750139 IC50 > 100000 nM T73184 CISM39 14119530 IC50 = 41500 nM T73184 CBX8T9 16451230 IC50 > 150000 nM T73184 CD8VI6 20088724 IC50 = 7200 nM T73184 CBL4S6 20232228 IC50 > 100000 nM T73184 C17HFK 22990729 IC50 = 42000 nM T73184 CJQ86Y 24827559 IC50 > 667000 nM T73184 C7S1QA 25216415 IC50 > 100000 nM T73184 CR8F9X 25218467 IC50 > 100000 nM T73184 C5N3LG 44251522 IC50 > 40000 nM T73184 CM8Z1G 53303486 IC50 = 9930 nM T73184 C70VHB 53315882 IC50 > 10000 nM T73184 CKAI31 53361222 IC50 = 174000 nM T73184 CV25JZ 53361223 IC50 = 149000 nM T73184 C0C6YK 53363652 IC50 > 667000 nM T73184 CPU86Z 53363653 IC50 > 667000 nM T73184 C63DVR 53363743 IC50 > 333000 nM T73184 COBL07 53363744 IC50 > 667000 nM T73184 C8QFS7 53363745 IC50 > 600000 nM T73184 CEG3P9 53363834 IC50 > 667000 nM T73184 CW4CD0 53363835 IC50 > 667000 nM T73184 CPL71I 54596764 IC50 = 49000 nM T73184 C2XR4C 56673504 IC50 = 66400 nM T73184 C04KFR 60150359 IC50 = 2200 nM T73184 CER5F1 67466175 IC50 = 214000 nM T73184 C4XJ5N 78357767 IC50 > 100000 nM T73184 CLU50V 122192598 IC50 = 89180 nM T73184 CA05IX 122192751 IC50 = 37670 nM T73184 C4U5VE 122192752 IC50 = 49520 nM T73184 CPKY06 122192761 IC50 = 61550 nM T73184 C2OU8A 127044062 IC50 > 100000 nM T73184 CU5Q0W 127044063 IC50 > 100000 nM T73184 CW0KT7 127045421 IC50 > 100000 nM T73184 C5ZM8O 137628302 IC50 > 100000 nM T73184 CW0C4P 155517779 IC50 > 100000 nM T73184 D00FLT 65482 IC50 = 2500 nM T73184 D02TVQ 71268957 IC50 = 63000 nM T73184 D09CLP 439155 IC50 = 30000 nM T73184 D0CX4W 46901937 IC50 > 40000 nM T73184 D0J6OV 71300326 Ki = 0.33 nM T47438 D00GPQ 46224413 IC50 = 1.2 nM T47438 D01LXD 9843750 IC50 = 38 nM T47438 D02HNG 9803433 IC50 = 5 nM T47438 D02JOH 46883536 IC50 = 0.13 nM T47438 D03MFQ 9996409 IC50 = 40000 nM T47438 D05FGR 92337 IC50 = 307000 nM T47438 D09ZVC 11269353 IC50 = 1.6 nM T47438 D0EV5O 46853593 EC50 = 29 nM T47438 D0F0JJ 11560787 IC50 = 64 nM T47438 D0I1OS 46854987 EC50 = 17 nM T47438 D0I3WC 49867930 IC50 = 4 nM T47438 D0O8UB 53241828 IC50 = 30 nM T47438 D0XI4P 91844660 IC50 = 7 nM T47438 D0D8IZ 25159185 IC50 = 8 nM T47438 D0K2YO 11964527 IC50 = 50 nM T47438 C40BXC 3803 IC50 = 30000 nM T47438 C19WAN 92803 EC50 = 5700 nM T47438 CA5BV8 169545 IC50 = 900 nM T47438 CQL19V 822847 IC50 = 1004 nM T47438 C5CG7L 965266 IC50 > 30000 nM T47438 CM73HW 2338583 IC50 > 40000 nM T47438 COK1Y6 2470340 IC50 > 40000 nM T47438 C0JR9A 2842595 IC50 = 2002 nM T47438 C5V6TP 3103157 IC50 = 2300 nM T47438 CK93HP 3844414 IC50 = 1540 nM T47438 C2B6AE 4788452 IC50 > 10000 nM T47438 CG5CH7 5155899 IC50 = 8278 nM T47438 C79BWF 5311272 IC50 = 500 nM T47438 CJ8P4T 5352624 IC50 = 53000 nM T47438 C0W3XG 5479543 IC50 = 17 nM T47438 CQ94WM 6324639 IC50 = 90 nM T47438 C76SLZ 7200833 IC50 = 966 nM T47438 CI8N0S 9805486 IC50 = 1 nM T47438 CPUY29 9807338 IC50 = 2.3 nM T47438 CI48QZ 9840950 IC50 = 651 nM T47438 CGSO64 9849380 IC50 = 5.6 nM T47438 C7TAZ2 9850372 IC50 = 17000 nM T47438 C3NF1M 9867067 IC50 = 0.19 nM T47438 C6KG4D 9874174 IC50 = 10 nM T47438 C0PN1K 9887090 IC50 = 491 nM T47438 CN3FH5 9893310 IC50 = 13.2 nM T47438 CIUM38 9901028 IC50 = 4408 nM T47438 C7Z5LV 9906160 IC50 = 70 nM T47438 CR91HS 9909323 IC50 = 32700 nM T47438 CHP82G 9910347 IC50 = 0.7 nM T47438 CD21QJ 9929326 IC50 = 3 nM T47438 C3KA5Q 9987560 IC50 = 70 nM T47438 COFE18 10002640 IC50 = 0.015 nM T47438 C0H1VQ 10117786 IC50 = 88 nM T47438 CWH3N7 10120043 IC50 = 56 nM T47438 C7ZR4N 10127574 IC50 = 570 nM T47438 CAQ5C6 10129054 IC50 = 8 nM T47438 CVX4J2 10143259 IC50 = 39 nM T47438 CXB8A6 10143260 IC50 = 540 nM T47438 C1M6SJ 10151615 IC50 = 6420 nM T47438 CLIO84 10163543 IC50 = 394 nM T47438 CU1A2J 10164752 IC50 = 2959 nM T47438 CG31VE 10175216 IC50 = 17 nM T47438 CR6LU7 10185072 IC50 = 299 nM T47438 CHL6W8 10194301 IC50 = 1970 nM T47438 C9MP6N 10194302 IC50 = 10620 nM T47438 CEV5A9 10196568 IC50 = 67 nM T47438 CPML95 10206761 IC50 = 504 nM T47438 C1AI8H 10227941 IC50 = 1096 nM T47438 CY7HG6 10239951 IC50 = 11 nM T47438 C2NU0D 10273953 IC50 = 4488 nM T47438 COQ19A 10277002 IC50 = 1644 nM T47438 C7FUL5 10311969 IC50 = 16 nM T47438 CG58VR 10341444 IC50 = 34200 nM T47438 C46JQA 10341445 IC50 = 24000 nM T47438 C9RE5W 10430137 IC50 = 22 nM T47438 CL3TN5 10434562 IC50 = 4.2 nM T47438 C0QNE9 10435235 EC50 = 0.119 nM T47438 CG2RL8 10459991 IC50 = 160 nM T47438 C2J6TA 10486685 IC50 = 780 nM T47438 CQ29TO 11062179 IC50 = 30000 nM T47438 CCR6J0 11152627 IC50 = 304 nM T47438 CN1L7M 11166476 IC50 = 400 nM T47438 C7LU4F 11169411 IC50 = 5000 nM T47438 C8SN4H 11169663 IC50 = 800 nM T47438 CTSQ29 11189908 IC50 = 230 nM T47438 C62ZWP 11192631 IC50 = 4000 nM T47438 C4CN2H 11193105 IC50 = 8000 nM T47438 CTP7N8 11226810 IC50 = 7000 nM T47438 CCD9V7 11240339 IC50 = 28 nM T47438 CJB5O8 11249248 IC50 = 7.1 nM T47438 CD8XH1 11250722 IC50 = 1000 nM T47438 CIDX13 11251926 IC50 = 9 nM T47438 CGZ49K 11257831 IC50 = 0.09 nM T47438 C3TV2Y 11273945 IC50 = 6000 nM T47438 C2F7MP 11285138 IC50 = 10 nM T47438 CTX52V 11297905 IC50 = 4700 nM T47438 CQ2P1S 11297908 IC50 = 26 nM T47438 CJ4R9F 11305056 IC50 = 0.024 nM T47438 CB9D7R 11306390 IC50 = 1 nM T47438 CWSA02 11319688 IC50 = 30 nM T47438 CJ6P7M 11329213 IC50 = 8.6 nM T47438 CL0GS1 11343941 IC50 = 14 nM T47438 C9LVZ8 11351105 IC50 = 3500 nM T47438 CQAS73 11366816 IC50 = 10000 nM T47438 CX8DT9 11366854 IC50 = 3100 nM T47438 C80KEI 11366911 IC50 = 910 nM T47438 C9S0MA 11376832 IC50 = 36.1 nM T47438 CHX4B9 11396006 IC50 = 0.042 nM T47438 CK3A1O 11423529 IC50 = 11000 nM T47438 CHW4L9 11430149 IC50 = 320 nM T47438 C63FEX 11431866 IC50 = 315 nM T47438 C7KLS0 11431964 IC50 = 76 nM T47438 CQ45UY 11454028 IC50 = 2.6 nM T47438 CW17SH 11456449 IC50 = 3000 nM T47438 CHZI35 11476771 IC50 = 76 nM T47438 C0TR9L 11479461 IC50 = 3000 nM T47438 C8WI9Y 11488357 IC50 = 100 nM T47438 CUO49D 11490643 IC50 = 60 nM T47438 CZ5JD8 11491881 IC50 = 16 nM T47438 CS6KW9 11494770 IC50 = 10 nM T47438 CL02TM 11503850 IC50 = 170 nM T47438 C2BI4M 11510496 IC50 = 9.1 nM T47438 CR71GB 11526691 IC50 = 9.9 nM T47438 C8YHU5 11548091 IC50 = 40 nM T47438 CR75FZ 11577204 IC50 = 15 nM T47438 C4BCJ3 11584234 IC50 = 6 nM T47438 CE9C5X 11596669 IC50 = 5 nM T47438 C6FAC1 11597267 IC50 = 80 nM T47438 CKDQ36 11627523 IC50 = 15 nM T47438 CQ75LF 11649620 IC50 = 20 nM T47438 C1ND2H 11697625 EC50 = 1258.93 nM T47438 C2LPQ8 11713496 IC50 = 120 nM T47438 C9Z6LE 11744162 IC50 = 5 nM T47438 CGTO42 11754136 IC50 = 10 nM T47438 C6Y8RF 11763616 IC50 = 800 nM T47438 CU2XG6 11815760 IC50 = 360 nM T47438 CYM80H 11817327 IC50 > 40000 nM T47438 CQ26XH 11851431 IC50 = 2.5 nM T47438 C0FSC7 11957110 IC50 = 0.06 nM T47438 C0YZH6 12147040 IC50 = 600 nM T47438 CQF06G 15071516 IC50 > 100000 nM T47438 C8WZH7 15208713 IC50 > 80000 nM T47438 C2D9TY 15344717 IC50 = 3100 nM T47438 C4VGL7 15767758 IC50 = 3000 nM T47438 CTM5I8 15942638 IC50 = 4 nM T47438 CA06DN 15953832 IC50 = 0.24 nM T47438 C6K8ZI 16035476 IC50 = 2 nM T47438 C7C2IK 16037832 IC50 = 3 nM T47438 CRT2F4 16043233 IC50 = 2.9 nM T47438 C8JZ4F 16043234 IC50 = 2000 nM T47438 CWD6X4 16045311 IC50 = 879 nM T47438 C7XPD5 16045393 IC50 = 151 nM T47438 CKOF24 16045394 IC50 = 6443 nM T47438 CSKY14 16045395 IC50 = 8 nM T47438 CWR7C1 16045555 IC50 = 26 nM T47438 CZB5M6 16085321 EC50 = 100 nM T47438 C9VPN2 16098384 EC50 = 20000 nM T47438 CCR68Z 16098385 EC50 > 20000 nM T47438 C51CIY 16098413 IC50 = 8500 nM T47438 C2WKD8 16098417 IC50 > 80000 nM T47438 CVYP36 16098434 IC50 > 40000 nM T47438 CPH4M3 16098435 IC50 = 2900 nM T47438 CP79WX 16112999 IC50 = 0.4 nM T47438 CSV24U 16655068 IC50 = 7500 nM T47438 C85AMK 16681308 IC50 = 21.2 nM T47438 CY1IH6 16722524 IC50 = 30 nM T47438 C70XVQ 16730389 IC50 = 598 nM T47438 CJ5YM2 16730390 IC50 = 80.9 nM T47438 CZW3O4 16730475 IC50 = 87 nM T47438 CAR4X1 16730476 IC50 = 5.4 nM T47438 C3XR6P 16730477 IC50 = 3.4 nM T47438 CF4LC6 16730478 IC50 = 776 nM T47438 CJ6YP9 16730566 IC50 = 536 nM T47438 C3BQ9R 16730567 IC50 = 120 nM T47438 C30OCW 16730568 IC50 = 10.2 nM T47438 CJ46CG 16730569 IC50 = 431 nM T47438 CODA06 16730724 IC50 = 244 nM T47438 CP30ZR 16730725 IC50 = 858 nM T47438 C7R1VI 16730727 IC50 > 40000 nM T47438 CC7QG9 16730799 IC50 = 350 nM T47438 C2PDT9 17747070 Ki = 2.6 nM T47438 CG3J5R 17747160 IC50 = 0.2 nM T47438 CAV2Z1 17986064 IC50 > 1000 nM T47438 C3G5ES 17986074 IC50 = 190 nM T47438 C0PRT8 17986076 IC50 = 7 nM T47438 CAN4I0 17986083 IC50 = 6000 nM T47438 C6MBD8 17986087 IC50 > 1000 nM T47438 C1RNQ6 17986094 IC50 > 1000 nM T47438 CK4RU9 17986184 IC50 = 70 nM T47438 CDC91U 18455128 IC50 = 1100 nM T47438 CVNB70 18455435 IC50 = 900 nM T47438 CLEI18 21048992 IC50 = 2.2 nM T47438 CS2EQ3 21049006 IC50 = 1.7 nM T47438 C3CL6R 21072502 IC50 = 3.3 nM T47438 C3CQZ6 21963897 IC50 = 4.2 nM T47438 CA48DB 21963931 IC50 = 1.4 nM T47438 C4YP3O 21963960 IC50 = 8.8 nM T47438 C38MFL 21963963 IC50 = 2.1 nM T47438 C6A7PO 21963967 IC50 = 21.5 nM T47438 CB18XR 21963968 IC50 = 148 nM T47438 CW3K9Z 21963972 IC50 = 14.3 nM T47438 CQH9L3 21963984 IC50 = 1.3 nM T47438 CO1UT3 21963988 IC50 = 1 nM T47438 CL74HI 22147970 IC50 = 1.65 nM T47438 C0A2BJ 22275595 IC50 = 40 nM T47438 CGF72V 22275717 IC50 = 2100 nM T47438 C15ZNF 22485769 IC50 = 510 nM T47438 C8LP1I 22984074 IC50 = 210 nM T47438 C32HUC 23028858 IC50 = 35 nM T47438 C05UKY 23509685 IC50 > 100000 nM T47438 CD6T3Z 23571062 IC50 = 0.06 nM T47438 CX1S4N 23571063 IC50 = 0.17 nM T47438 CYS7G4 23571064 IC50 = 0.42 nM T47438 C3GVY5 23571065 IC50 = 0.12 nM T47438 CU6IF5 23571066 IC50 = 0.82 nM T47438 CIBK15 23571067 IC50 = 0.08 nM T47438 C5T1SC 23571069 IC50 = 0.15 nM T47438 CXQ8R3 23571070 IC50 = 0.03 nM T47438 CC6N9Y 23571085 IC50 = 0.06 nM T47438 C68MVY 23571092 IC50 = 0.41 nM T47438 C06ZKN 23571093 IC50 = 0.06 nM T47438 CEPG49 23571096 IC50 = 0.07 nM T47438 CF7X5B 23571100 IC50 = 0.42 nM T47438 CB1R2P 23571105 IC50 = 0.34 nM T47438 C94OLI 23571205 IC50 = 0.21 nM T47438 C09CFT 23590946 IC50 = 4.7 nM T47438 CQ0JA6 23590952 IC50 = 0.51 nM T47438 CX36KQ 23627219 IC50 = 27 nM T47438 CNT92F 23656215 IC50 = 0.3 nM T47438 CIT4M2 23661615 IC50 = 7.8 nM T47438 CCX9Y5 23661672 IC50 = 5 nM T47438 CP93XI 23661699 IC50 = 2.4 nM T47438 CE5QD9 24180447 IC50 = 19600 nM T47438 C6FM9C 24180452 IC50 = 6.9 nM T47438 CB7ZC2 24180609 IC50 = 93 nM T47438 CK71ZR 24767800 IC50 = 2700 nM T47438 C8G7JD 24768566 IC50 = 96000 nM T47438 C3AM6Z 24779751 IC50 = 4.4 nM T47438 C03HRN 24864172 IC50 = 22 nM T47438 CE8DS6 24864173 IC50 = 220 nM T47438 CCX4P2 24864336 IC50 = 1.2 nM T47438 CK6E5Q 24864337 IC50 = 2 nM T47438 CVRN07 24864341 IC50 = 290 nM T47438 CG5CA4 24864523 IC50 = 1.6 nM T47438 C1V7WL 24864526 IC50 = 0.74 nM T47438 CIXE60 24864527 IC50 = 140 nM T47438 CDOV21 24864705 IC50 = 0.36 nM T47438 CK17JW 24864708 IC50 = 1.4 nM T47438 C8L0RO 24864709 IC50 = 2.1 nM T47438 CJ64HZ 24864711 IC50 = 0.17 nM T47438 CHG7C1 24864885 IC50 = 0.21 nM T47438 CREF30 24864886 IC50 = 0.28 nM T47438 CK2R6U 24865064 IC50 = 0.93 nM T47438 CJ1I9X 24865066 IC50 = 4.5 nM T47438 CGJ2Q4 24865068 IC50 = 2.6 nM T47438 CQ24JB 24865069 IC50 = 27 nM T47438 C1XP9G 24865249 IC50 = 0.52 nM T47438 CM17UV 24865251 IC50 = 1.1 nM T47438 CR8DV9 24865253 IC50 = 0.42 nM T47438 C26BIY 24865786 IC50 = 1.3 nM T47438 CN7GO5 24865789 IC50 = 2.4 nM T47438 C3HE0S 24865989 IC50 = 280 nM T47438 CSID98 24865993 IC50 = 85 nM T47438 C7I4VC 24866171 IC50 = 40 nM T47438 C48OQZ 24866173 IC50 = 0.46 nM T47438 CY0UC2 24866175 IC50 = 2.1 nM T47438 CZ1O3X 24866342 IC50 = 0.76 nM T47438 CE1FY8 24866343 IC50 = 5500 nM T47438 CP40OT 24866346 IC50 = 24 nM T47438 C8C5JG 24896257 IC50 = 5.6 nM T47438 C79GSB 24936138 IC50 = 0.32 nM T47438 C0B5LM 24936139 IC50 = 5.6 nM T47438 CKYX49 24963625 IC50 = 880 nM T47438 CU38IK 24964342 IC50 = 710 nM T47438 CQ7UB1 24964343 IC50 = 230 nM T47438 CXE6Q3 24964696 IC50 = 490 nM T47438 CWO1V4 25004449 IC50 = 840 nM T47438 CJR3M7 25014542 IC50 = 15000 nM T47438 CZ7G9O 25024968 IC50 = 28840 nM T47438 C5C7KU 25025157 IC50 > 50000 nM T47438 CG8WN5 25032613 IC50 = 0.27 nM T47438 C86CQY 25052759 IC50 = 214 nM T47438 CP7MH1 25106114 IC50 = 339 nM T47438 C98CGM 25106115 IC50 = 136 nM T47438 CLD7X0 25107258 IC50 = 898 nM T47438 C4NE6H 25107259 IC50 = 880 nM T47438 COT5G4 25107260 IC50 = 789 nM T47438 CL4XY0 25125138 IC50 = 2770 nM T47438 CIYA24 25125139 IC50 = 440 nM T47438 CH6Q5L 25125140 IC50 = 1440 nM T47438 C56EUJ 25138385 IC50 = 11 nM T47438 CW3OC1 25143875 IC50 = 58 nM T47438 C3DY8R 25144288 IC50 = 15 nM T47438 C2H4KJ 25145553 IC50 = 58 nM T47438 C3SOU5 25145846 IC50 = 75 nM T47438 CTF47W 25164607 IC50 = 1.3 nM T47438 CLW81T 25164608 IC50 = 7.4 nM T47438 CTB5M4 25164609 IC50 = 2 nM T47438 CQK4J3 25164810 IC50 = 6.4 nM T47438 CIJ2P5 25164811 IC50 = 6.8 nM T47438 CEKW51 25164812 IC50 = 5.5 nM T47438 C76DCT 25165012 IC50 = 25 nM T47438 C51XTP 25165014 IC50 = 0.9 nM T47438 C4ZJQ7 25165409 IC50 = 2.9 nM T47438 C3OIX5 25165410 IC50 = 1.4 nM T47438 CIXD52 25165995 IC50 = 63 nM T47438 C87EJY 25166594 IC50 = 5100 nM T47438 CVW64A 25166800 IC50 = 360 nM T47438 CSMD23 25186150 IC50 = 56 nM T47438 C52CEB 25186926 IC50 = 2 nM T47438 C2CTD9 25187263 IC50 = 135 nM T47438 CJL7I6 25225345 IC50 = 446 nM T47438 C82QUJ 25255222 IC50 = 144 nM T47438 CYOM53 25255427 IC50 = 94 nM T47438 C8TU1B 25255724 IC50 = 139 nM T47438 CD2GN0 25256437 IC50 = 322 nM T47438 CHP5E1 25256439 IC50 = 864 nM T47438 C4LMN1 25256522 IC50 = 955 nM T47438 C6J2PH 25256523 IC50 = 671 nM T47438 CO91CG 25263468 IC50 = 1 nM T47438 C4J1HV 25263469 IC50 = 0.65 nM T47438 C47ASX 25263470 IC50 = 0.51 nM T47438 CG4AI6 25263471 IC50 = 1.1 nM T47438 C83NHE 25263472 IC50 = 0.36 nM T47438 CKD1S7 25263473 IC50 = 1.9 nM T47438 CBY15W 25263474 IC50 = 35 nM T47438 CZ0TO9 25263475 IC50 = 0.82 nM T47438 CN65HK 25263476 IC50 = 0.25 nM T47438 C6Q5GS 25263477 IC50 = 0.66 nM T47438 C74ACU 25263478 IC50 = 0.15 nM T47438 C7RD5S 25263479 IC50 = 15 nM T47438 CP96SY 25263480 IC50 = 10 nM T47438 CW74XQ 25263481 IC50 = 2.1 nM T47438 CZ40XH 25263482 IC50 = 12 nM T47438 CT2MI1 25263483 IC50 = 15 nM T47438 CQL04P 25263484 IC50 = 12 nM T47438 CX3N1M 25263485 IC50 = 18 nM T47438 CRI45P 25263486 IC50 = 1.8 nM T47438 CC2FN6 25263487 IC50 = 0.93 nM T47438 CSKO45 25263488 IC50 = 4 nM T47438 CFH95Q 25263489 IC50 = 7.7 nM T47438 COIC78 25263490 IC50 = 0.06 nM T47438 C74LDY 25263491 IC50 = 0.06 nM T47438 C1WL7C 25263492 IC50 = 19 nM T47438 CIJU03 25263493 IC50 = 1.2 nM T47438 CF61JK 25263494 IC50 = 0.66 nM T47438 CP4TF9 25263495 IC50 = 0.41 nM T47438 CGO2Q4 25263496 IC50 = 0.48 nM T47438 CYG7A3 25263497 IC50 = 0.51 nM T47438 CZ2T1W 42632633 IC50 = 50.12 nM T47438 CZR8L4 42632635 IC50 = 63.1 nM T47438 C67ZYN 42632637 IC50 = 50.12 nM T47438 CS95DW 42632653 IC50 = 63.1 nM T47438 CM8OV5 42632655 IC50 = 199.53 nM T47438 CSGK56 42632682 IC50 = 316.23 nM T47438 CXD8G0 42632750 IC50 = 199.53 nM T47438 C5QE0V 42632752 IC50 = 630.96 nM T47438 C05NRU 42632754 IC50 = 158.49 nM T47438 CEVN24 42632772 IC50 = 316.23 nM T47438 CT8L3J 42632842 IC50 = 125.89 nM T47438 C6NZ5A 42632900 IC50 = 125.89 nM T47438 C87POD 42633502 IC50 = 116 nM T47438 CAX43F 42633863 IC50 = 509 nM T47438 C0S8GC 42638432 IC50 = 500 nM T47438 CZS65J 42638433 IC50 = 1200 nM T47438 CH3MY1 42639933 IC50 = 260 nM T47438 CVY8H2 42640092 IC50 = 460 nM T47438 CU68PM 42640420 IC50 = 170 nM T47438 CRGV67 42640423 IC50 = 540 nM T47438 CT0OU1 42640598 IC50 = 2780 nM T47438 C2MY8X 42647277 IC50 = 44 nM T47438 CX3L0P 44139437 IC50 = 8.81 nM T47438 C3ZGR9 44157625 IC50 = 0.46 nM T47438 CA9FN6 44193857 IC50 = 209 nM T47438 CE5A9Z 44193858 IC50 = 133 nM T47438 CFEX37 44193859 IC50 = 244 nM T47438 CBC3W9 44193860 IC50 = 252 nM T47438 C19RXP 44193960 IC50 = 212 nM T47438 CEM1J3 44193962 IC50 = 127 nM T47438 CU06VM 44193963 IC50 = 651 nM T47438 CE1PW4 44194155 IC50 = 319 nM T47438 CBS1D6 44195184 IC50 = 133 nM T47438 C5T3FW 44195186 IC50 = 123 nM T47438 CV6WM1 44241633 IC50 = 154 nM T47438 C3SFT9 44272269 IC50 = 5000 nM T47438 CA4F7H 44272270 IC50 = 3400 nM T47438 C7EQ2R 44272404 IC50 = 400 nM T47438 CL15MO 44272482 IC50 = 15000 nM T47438 CL4J3Z 44272483 IC50 = 180 nM T47438 C6L1IY 44272484 IC50 = 400 nM T47438 CS67FV 44272499 IC50 = 1500 nM T47438 CQHE15 44272500 IC50 = 1600 nM T47438 CK5EV7 44272502 IC50 = 550 nM T47438 C3HB6A 44272553 IC50 = 580 nM T47438 CP3NY6 44272576 IC50 = 620 nM T47438 C81DBR 44272577 IC50 = 15000 nM T47438 C0ME2L 44272578 IC50 = 450 nM T47438 CQYN68 44272595 IC50 = 300 nM T47438 C48XAS 44272596 IC50 = 17000 nM T47438 C9W6EG 44272620 IC50 > 25000 nM T47438 C8DG3U 44272639 IC50 > 25000 nM T47438 CTJ28F 44272794 IC50 > 25000 nM T47438 C6I7FY 44272815 IC50 = 3300 nM T47438 CA5C6N 44272822 IC50 = 600 nM T47438 C1ARU0 44272823 IC50 = 900 nM T47438 C79FBO 44272863 IC50 = 920 nM T47438 CL0PB6 44272874 IC50 = 1800 nM T47438 CL08UE 44299780 IC50 = 1200 nM T47438 CIMP62 44299785 IC50 = 240 nM T47438 CTP4K5 44299806 IC50 = 150 nM T47438 CFDX15 44299807 IC50 = 800 nM T47438 CO58LY 44299816 IC50 = 1100 nM T47438 C72ICU 44299831 IC50 = 6 nM T47438 CD4K9L 44299838 IC50 = 480 nM T47438 C4JC6H 44299839 IC50 = 4.7 nM T47438 CB9W1F 44299856 IC50 > 2500 nM T47438 CI8H6V 44299857 IC50 = 454 nM T47438 CSBE57 44299884 IC50 = 1000 nM T47438 CD7K6U 44299900 IC50 > 2500 nM T47438 C4IB5Y 44299922 IC50 = 20 nM T47438 CQIZ85 44299941 IC50 = 408 nM T47438 CCZ5H7 44299970 IC50 = 3200 nM T47438 C8AJ3U 44299981 IC50 = 240 nM T47438 CEBH91 44299982 IC50 > 2600 nM T47438 CO26SB 44299986 IC50 = 160 nM T47438 C34TQN 44299987 IC50 = 71 nM T47438 C72LXP 44300008 IC50 = 1700 nM T47438 C9JUG3 44300019 IC50 > 2500 nM T47438 CHV7K8 44300020 IC50 = 66 nM T47438 C06ZXT 44300027 IC50 > 2500 nM T47438 C45QVN 44300045 IC50 = 300 nM T47438 CD6VT9 44300046 IC50 = 32 nM T47438 CH3BD1 44300054 IC50 > 2500 nM T47438 C37NVU 44300062 IC50 = 2400 nM T47438 C9B4TQ 44300116 IC50 = 280 nM T47438 C3G7CU 44300117 IC50 = 900 nM T47438 CDUB40 44300118 IC50 = 800 nM T47438 C1MW5E 44300137 IC50 = 50 nM T47438 C6IAU4 44300141 IC50 = 102 nM T47438 C43QHF 44300156 IC50 = 55 nM T47438 C6OT5P 44300185 IC50 = 52 nM T47438 CZX60N 44300200 IC50 = 36 nM T47438 C4F9SV 44300201 IC50 > 2500 nM T47438 CU82ZK 44300204 IC50 > 2500 nM T47438 CW3M8K 44300206 IC50 > 2500 nM T47438 C1C0FH 44300213 IC50 > 2500 nM T47438 CM5Y2D 44300220 IC50 > 2500 nM T47438 C04MOF 44300225 IC50 = 2000 nM T47438 CEFA26 44300242 IC50 = 1 nM T47438 CFJ3S7 44300372 IC50 > 2500 nM T47438 CPKU38 44300560 IC50 = 300 nM T47438 CKE03P 44300566 IC50 = 13 nM T47438 CDJ1K4 44300571 IC50 = 130 nM T47438 CZ29RH 44300582 IC50 = 39 nM T47438 CMOE73 44300584 IC50 = 17 nM T47438 C8CT2N 44344777 IC50 = 140 nM T47438 CAK7D0 44344792 IC50 = 57 nM T47438 CA6G8L 44344798 IC50 = 720 nM T47438 CMV09U 44344902 IC50 > 2500 nM T47438 CVH04W 44344916 IC50 = 5 nM T47438 C3S7ZH 44344917 IC50 = 14 nM T47438 C4KUV7 44344918 IC50 = 38 nM T47438 CPZ1M7 44344923 IC50 = 86 nM T47438 CM4FQ2 44344936 IC50 > 2500 nM T47438 C4L6GK 44344979 IC50 = 47 nM T47438 CG3TN7 44344993 IC50 = 1500 nM T47438 C4YU7O 44345078 IC50 = 4 nM T47438 CTD02F 44345083 IC50 = 37 nM T47438 CJ0R9G 44345100 IC50 = 190 nM T47438 CBQ50F 44345133 IC50 = 150 nM T47438 CHZ46Y 44345144 IC50 > 2500 nM T47438 CXPR42 44345153 IC50 > 2500 nM T47438 CI7B2O 44345154 IC50 > 2500 nM T47438 C2OE7B 44354160 IC50 = 1884 nM T47438 C93ODM 44354173 IC50 = 100.6 nM T47438 C72GNU 44354186 IC50 = 4.7 nM T47438 C4IL1K 44354199 IC50 = 2.2 nM T47438 C0ICU7 44354337 IC50 = 5.5 nM T47438 C93ZCV 44354338 IC50 = 28 nM T47438 CJPT35 44354363 IC50 = 12.7 nM T47438 C6FDY5 44354364 IC50 = 1.8 nM T47438 CSFK05 44354431 IC50 = 0.49 nM T47438 CIF9Q4 44354432 IC50 = 0.9 nM T47438 CMG1C8 44354433 IC50 = 3.7 nM T47438 CSM8K2 44354444 IC50 = 13.2 nM T47438 CGJU57 44354445 IC50 = 1.2 nM T47438 CQY1M8 44354459 IC50 = 1.8 nM T47438 C0VL9I 44354463 IC50 = 3.6 nM T47438 CD02RP 44354512 IC50 = 0.3 nM T47438 CK2I9B 44386459 IC50 = 400 nM T47438 C0K1RP 44386460 IC50 = 390 nM T47438 C1DIV7 44386461 IC50 = 18000 nM T47438 C5Q8HR 44386506 IC50 = 230 nM T47438 C97HRQ 44386664 IC50 = 8000 nM T47438 CB7C4E 44386766 IC50 = 20000 nM T47438 CE6Y3A 44386767 IC50 = 250 nM T47438 CQ4LM3 44386768 IC50 = 150 nM T47438 CC0MF8 44386780 IC50 = 22000 nM T47438 CZ51MR 44386781 IC50 = 400 nM T47438 C4TY6U 44386828 IC50 = 140 nM T47438 CU9TH3 44386902 IC50 = 500 nM T47438 C0NRO6 44387006 IC50 = 670 nM T47438 CBHG04 44387127 IC50 = 530 nM T47438 C67JZV 44387228 IC50 = 540 nM T47438 C7J2SN 44388746 IC50 = 152 nM T47438 CLY7C6 44388755 IC50 = 623 nM T47438 C1LJ6O 44388757 IC50 = 39 nM T47438 CE85NT 44388765 IC50 = 335 nM T47438 CQL81R 44388767 IC50 = 21 nM T47438 C8RJW0 44388774 IC50 = 15 nM T47438 C4F3XD 44388775 IC50 = 209 nM T47438 C4OS5H 44388781 IC50 = 5 nM T47438 CSD0H2 44391778 IC50 > 1000 nM T47438 CCTX25 44391779 IC50 = 62 nM T47438 CMD12V 44391780 IC50 = 29 nM T47438 CW1M4K 44391785 IC50 > 1000 nM T47438 C56HFN 44391787 IC50 = 16 nM T47438 CH0YT8 44391790 IC50 > 1000 nM T47438 CGZ06W 44391795 IC50 = 75 nM T47438 CX1Z5Y 44391797 IC50 > 1000 nM T47438 CEJ6X3 44391801 IC50 = 6 nM T47438 C9WSN6 44391803 IC50 > 1000 nM T47438 CPM3E0 44391804 IC50 = 721 nM T47438 CKD81U 44391806 IC50 = 34 nM T47438 C17PFC 44391809 IC50 = 239 nM T47438 CJT3D5 44391810 IC50 = 12 nM T47438 C1VP5T 44391812 IC50 = 146 nM T47438 C9N8MZ 44391813 IC50 = 412 nM T47438 CA5H3N 44391817 IC50 = 535 nM T47438 CR3D5J 44391818 IC50 = 7 nM T47438 C7HL9Y 44391819 IC50 = 610 nM T47438 C6ZJW2 44391822 IC50 = 324 nM T47438 CA59PK 44391823 IC50 > 1000 nM T47438 CQ23WT 44391825 IC50 = 175 nM T47438 CMQ25A 44391827 IC50 = 129 nM T47438 C3O7NC 44391829 IC50 = 153 nM T47438 C7KX2F 44391831 IC50 > 1000 nM T47438 CY45WQ 44391832 IC50 = 41 nM T47438 CX68DF 44391834 IC50 = 490 nM T47438 C9KPT6 44391836 IC50 > 1000 nM T47438 C6OD3B 44391837 IC50 = 269 nM T47438 CC0N5Q 44391839 IC50 > 1000 nM T47438 CVM40E 44391840 IC50 = 74 nM T47438 CP6A0L 44391845 IC50 = 69 nM T47438 COMI50 44391846 IC50 > 1000 nM T47438 CL8IU7 44391850 IC50 > 1000 nM T47438 C2GL0H 44391851 IC50 = 467 nM T47438 CM5G8L 44391852 IC50 = 23 nM T47438 CLT4I7 44391857 IC50 > 1000 nM T47438 CVOC09 44391862 IC50 = 3490 nM T47438 C0U6SQ 44391880 IC50 = 73 nM T47438 CR95TU 44391894 IC50 = 227 nM T47438 CGC76F 44391900 IC50 = 5 nM T47438 CT9N4H 44391911 IC50 = 226 nM T47438 CS19FK 44396232 IC50 = 25 nM T47438 C2ZVO0 44400673 IC50 = 12 nM T47438 C1K2IX 44400710 IC50 = 104 nM T47438 CUSQ68 44400771 IC50 = 170 nM T47438 C7Z5DM 44400772 IC50 = 27 nM T47438 C10QIO 44400790 IC50 = 55 nM T47438 C4V0IG 44400842 IC50 = 253 nM T47438 CTFY61 44400878 IC50 = 98 nM T47438 C8SO5T 44400879 IC50 = 1900 nM T47438 CPVJ60 44400904 IC50 = 2472 nM T47438 C4DBM3 44400933 IC50 = 249 nM T47438 C75GIF 44403333 IC50 = 62 nM T47438 C1UJK7 44403341 IC50 = 132 nM T47438 CGMY50 44403342 IC50 = 1 nM T47438 C3Y5PS 44403401 IC50 = 394 nM T47438 C89GRJ 44403409 IC50 = 766 nM T47438 CTC17R 44403410 IC50 = 134 nM T47438 C9ZSM3 44403413 IC50 = 429 nM T47438 CDA16M 44403414 IC50 = 138 nM T47438 C9Z2TM 44403415 IC50 = 122 nM T47438 CJSH92 44403418 IC50 = 17 nM T47438 C0YSJ9 44403419 IC50 = 19 nM T47438 C7TYW4 44403423 IC50 = 2 nM T47438 CY61LD 44403424 IC50 = 3.4 nM T47438 COVL82 44403428 IC50 = 250 nM T47438 CMZ25N 44403431 IC50 = 18 nM T47438 C7XJ8T 44403432 IC50 = 21 nM T47438 CK09NJ 44403434 IC50 = 4 nM T47438 CF7LQ4 44411586 IC50 = 1.39 nM T47438 CJA03K 44411650 IC50 = 0.24 nM T47438 CXG72Q 44411651 IC50 = 0.76 nM T47438 CPTX52 44411690 IC50 = 0.04 nM T47438 C2OS3K 44411691 IC50 = 0.08 nM T47438 CP9T4I 44411692 IC50 = 0.06 nM T47438 CY9BW4 44412059 IC50 = 0.4 nM T47438 CCD8N4 44412061 IC50 = 1.17 nM T47438 CH0O5Z 44412062 IC50 = 0.41 nM T47438 C79ZOD 44412080 IC50 = 0.19 nM T47438 C30DSF 44412081 IC50 = 0.9 nM T47438 C6HDY0 44412083 IC50 = 0.26 nM T47438 CMNE06 44412297 IC50 = 6.18 nM T47438 C85GSO 44413510 IC50 > 100000 nM T47438 CDM4F2 44413568 IC50 > 100000 nM T47438 C13BKF 44413569 IC50 = 500 nM T47438 C58TNH 44413653 IC50 = 85 nM T47438 C26HYC 44413654 IC50 = 8 nM T47438 CJ4U8X 44413659 IC50 > 100000 nM T47438 CJXW54 44413660 IC50 = 4600 nM T47438 C0K8UY 44413669 IC50 = 112 nM T47438 C4X5BG 44413670 IC50 = 24 nM T47438 CFU14K 44413689 IC50 = 380 nM T47438 CZ3B4H 44413690 IC50 = 10 nM T47438 CG5N4R 44413701 IC50 = 210 nM T47438 CB52ER 44413711 IC50 = 44 nM T47438 CDG6W4 44413753 IC50 = 1628 nM T47438 C4TZ7D 44413785 IC50 = 7200 nM T47438 CL7Y8W 44413786 IC50 = 5900 nM T47438 C8HUB4 44413791 IC50 = 376 nM T47438 CM6D4R 44413792 IC50 = 77 nM T47438 C21BHJ 44413797 IC50 > 100000 nM T47438 CAV8Z0 44413798 IC50 = 26000 nM T47438 C87MVI 44413804 IC50 = 55 nM T47438 CW8CK0 44413805 IC50 = 10 nM T47438 CQ4NY3 44413810 IC50 > 100000 nM T47438 CJP10D 44413812 IC50 > 100000 nM T47438 CTM24D 44413821 IC50 > 100000 nM T47438 C1O3DB 44413822 IC50 > 100000 nM T47438 C0PZ4N 44414662 IC50 = 1000 nM T47438 C60SKV 44414672 IC50 = 1100 nM T47438 C6GV4A 44414676 IC50 = 130 nM T47438 CN0S8T 44414677 IC50 = 17000 nM T47438 CW73JT 44414685 IC50 = 490 nM T47438 C4JD8U 44414686 IC50 = 10 nM T47438 C3U0HO 44414698 IC50 = 530 nM T47438 C7Z2DP 44414744 IC50 = 3200 nM T47438 CEVF60 44414745 IC50 = 10 nM T47438 C6PA2W 44414746 IC50 = 20 nM T47438 C96UKI 44414773 IC50 = 4400 nM T47438 CJ3H8L 44414774 IC50 = 1300 nM T47438 CX15LW 44414778 IC50 = 6.1 nM T47438 CF3E7Y 44414797 IC50 = 470 nM T47438 CNI3J4 44414807 IC50 = 530 nM T47438 C8LKZ2 44414808 IC50 = 350 nM T47438 CG4MU6 44414826 IC50 = 400 nM T47438 CKHW96 44414838 IC50 = 1900 nM T47438 CM68NQ 44414839 IC50 = 690 nM T47438 C5HG7K 44414857 IC50 = 1200 nM T47438 CLSE91 44414858 IC50 = 3000 nM T47438 C1AGV6 44421238 IC50 = 200 nM T47438 CCKQ89 44421239 IC50 = 7000 nM T47438 C7BA5U 44421240 IC50 = 2000 nM T47438 CPY82H 44421241 IC50 = 3000 nM T47438 C9VH0I 44421242 IC50 = 3000 nM T47438 CO9XG3 44421243 IC50 = 2000 nM T47438 CF64CH 44421244 IC50 = 24000 nM T47438 C2ACK0 44421245 IC50 = 12000 nM T47438 C6PXS2 44421246 IC50 = 3000 nM T47438 CG7V9P 44421321 IC50 = 900 nM T47438 CADE57 44421322 IC50 = 2000 nM T47438 CL13AF 44421323 IC50 = 6000 nM T47438 C6G0XP 44421334 IC50 = 5000 nM T47438 C9R0TM 44421335 IC50 = 600 nM T47438 CCJB73 44429704 IC50 = 2500 nM T47438 CM6GO3 44429705 IC50 = 680 nM T47438 C46SOY 44429706 IC50 = 270 nM T47438 CHR0P6 44429707 IC50 = 15420 nM T47438 C1I2WC 44429708 IC50 = 219 nM T47438 C3MLB9 44429709 IC50 = 159 nM T47438 CDOV06 44429710 IC50 = 34 nM T47438 C73NZY 44429711 IC50 = 12300 nM T47438 CL23CT 44429712 IC50 = 4770 nM T47438 CNEI43 44429713 IC50 = 71 nM T47438 CUK8Q2 44429715 IC50 = 37 nM T47438 C2CB3A 44429716 IC50 = 38 nM T47438 C73HBA 44429717 IC50 = 26 nM T47438 C9I5KO 44429718 IC50 = 13 nM T47438 C0XP3E 44429723 IC50 = 28 nM T47438 C83NCX 44429724 IC50 = 10 nM T47438 CE8U1T 44429726 IC50 = 36 nM T47438 CUQ1P7 44429727 IC50 = 7 nM T47438 CHZY93 44429728 IC50 = 4 nM T47438 CQ5WV3 44429729 IC50 = 26 nM T47438 C71IMA 44429730 IC50 = 8 nM T47438 C9ZGA2 44432541 Ki = 1000 nM T47438 CW2GR3 44432543 Ki = 227 nM T47438 CFWE67 44432548 Ki = 15 nM T47438 CS4BO0 44432549 Ki = 11 nM T47438 CDE85L 44432550 Ki = 3.5 nM T47438 C4JO5H 44432551 Ki = 1.2 nM T47438 C6ZF0L 44432552 Ki = 1.4 nM T47438 CGH6N0 44432554 Ki = 6.2 nM T47438 C4H9BC 44432556 Ki = 2 nM T47438 CC5L7X 44432557 Ki = 3 nM T47438 CK52RJ 44432568 IC50 = 19 nM T47438 CV3FY9 44432569 Ki = 36 nM T47438 C6G2BA 44432572 Ki = 9.9 nM T47438 C36YRT 44432575 Ki = 13.5 nM T47438 CY6CL0 44432578 Ki = 4.9 nM T47438 CM3DJ5 44432579 Ki = 4 nM T47438 C6KUW0 44432584 Ki = 2.2 nM T47438 CE1W6U 44432588 Ki = 1.3 nM T47438 CP24YK 44432590 Ki = 1.1 nM T47438 C89PTY 44432592 Ki = 3.9 nM T47438 C67PIK 44432596 Ki = 2.1 nM T47438 CE8US0 44432598 Ki = 0.9 nM T47438 CMA4O9 44432601 Ki = 22 nM T47438 C4DR0K 44432604 Ki = 3.1 nM T47438 C3XBU0 44432607 Ki = 111 nM T47438 CD0ET2 44432735 IC50 = 850 nM T47438 CH73FO 44432736 IC50 = 1100 nM T47438 CJY57U 44432737 IC50 = 750 nM T47438 C2SYG0 44432738 IC50 = 1300 nM T47438 C8FGR3 44432739 IC50 = 400 nM T47438 CDW4U1 44432740 IC50 = 700 nM T47438 C4I3RA 44432741 IC50 = 2000 nM T47438 C92DVC 44432742 IC50 = 920 nM T47438 CUC3O6 44432743 IC50 = 1000 nM T47438 CQ6G1T 44432744 IC50 = 350 nM T47438 CM17EH 44432745 IC50 = 190 nM T47438 C4FC1D 44432746 IC50 = 1000 nM T47438 C7QP9I 44432747 IC50 = 1200 nM T47438 CIJ31A 44432748 IC50 = 360 nM T47438 CU4LA7 44432749 IC50 = 720 nM T47438 CR78GI 44432750 IC50 = 1200 nM T47438 C5MR7Y 44432751 IC50 = 66 nM T47438 CIR93O 44432752 IC50 = 56 nM T47438 C2SUF9 44432753 IC50 = 19 nM T47438 C7GUX6 44432754 IC50 = 72 nM T47438 CLP08T 44432755 IC50 = 180 nM T47438 CSM3Y2 44432757 IC50 = 1300 nM T47438 CY2OV0 44432758 IC50 = 240 nM T47438 C6E1LT 44432759 IC50 = 560 nM T47438 CZKR96 44432760 IC50 > 25000 nM T47438 CFL9M6 44432780 IC50 = 13 nM T47438 C39CUV 44432782 IC50 = 140 nM T47438 CTZ64S 44432784 IC50 = 23 nM T47438 CQ1UV3 44432785 IC50 = 25 nM T47438 CT2JH3 44432787 IC50 = 7 nM T47438 CNC96Y 44432789 IC50 = 49 nM T47438 CK70ES 44432792 IC50 = 12 nM T47438 CNFB80 44432793 IC50 = 14 nM T47438 C06KEF 44432796 IC50 = 33 nM T47438 C68JBI 44432797 IC50 = 22 nM T47438 CNQ2X3 44432799 IC50 = 41 nM T47438 C4DHY0 44432800 IC50 = 100 nM T47438 CG7MS6 44432801 IC50 = 140 nM T47438 C80GXR 44432802 IC50 = 1300 nM T47438 CK5IO0 44432804 IC50 = 100 nM T47438 CN21WE 44432805 IC50 = 3700 nM T47438 CTZD96 44432807 IC50 = 24 nM T47438 CV4GI8 44432808 IC50 = 14 nM T47438 C1Z9UG 44432809 IC50 = 4 nM T47438 CV9AI5 44432810 IC50 = 5 nM T47438 C7PEV0 44433881 IC50 = 1500 nM T47438 C7JQW3 44433888 IC50 = 3.1 nM T47438 CZ8K2R 44433889 IC50 = 580 nM T47438 CNKB48 44433891 IC50 = 1.6 nM T47438 CCGZ80 44433893 IC50 = 7.1 nM T47438 CZ8G4V 44433896 IC50 = 5.3 nM T47438 CH0PB4 44433897 IC50 = 6.3 nM T47438 CE1BP2 44433898 IC50 = 12 nM T47438 C7TD8Q 44433899 IC50 = 22 nM T47438 CP19WA 44433901 IC50 = 20 nM T47438 CC76FQ 44433923 IC50 = 0.002 nM T47438 C7HSE9 44433930 IC50 = 1.7 nM T47438 C4Q2MH 44435366 IC50 = 27 nM T47438 CX51JK 44435367 IC50 = 12 nM T47438 C1SCL8 44435394 IC50 = 11.6 nM T47438 CVF83U 44435448 IC50 = 0.3 nM T47438 CO16ME 44435449 IC50 = 0.3 nM T47438 CT3NY9 44435450 IC50 = 7.49 nM T47438 C4CBZ6 44435451 IC50 = 0.05 nM T47438 C2TX3S 44435452 IC50 = 0.14 nM T47438 C4PM7B 44435453 IC50 = 30 nM T47438 C3UA0C 44435454 IC50 = 81.5 nM T47438 C54DVE 44435455 IC50 = 0.22 nM T47438 CW1O9L 44435456 IC50 = 0.22 nM T47438 CJO6U3 44435457 IC50 = 0.43 nM T47438 COB67F 44435458 IC50 = 0.11 nM T47438 CK84MV 44435459 IC50 = 1.14 nM T47438 C92MHT 44435460 IC50 = 50.5 nM T47438 C6PHM1 44435462 IC50 = 63.2 nM T47438 CWZ10L 44435463 IC50 = 42 nM T47438 C0QIS7 44435464 IC50 = 4.5 nM T47438 CY2V0F 44435465 IC50 = 10.1 nM T47438 C94BOF 44435466 IC50 = 29.8 nM T47438 C97KQX 44435467 IC50 = 2 nM T47438 C9U6ZV 44435468 IC50 = 7.1 nM T47438 CI4R2T 44435469 IC50 = 4.2 nM T47438 C3R4SW 44435470 IC50 = 3.1 nM T47438 CZ4L1H 44435471 IC50 = 134 nM T47438 CWF51G 44435472 IC50 = 2.6 nM T47438 CO17MG 44435473 IC50 = 5 nM T47438 CMVY01 44435474 IC50 = 2.7 nM T47438 CO7PI4 44435475 IC50 = 5.9 nM T47438 CBG0P2 44435476 IC50 = 28.3 nM T47438 C7VGP3 44435477 IC50 = 1.4 nM T47438 CKJV32 44435478 IC50 = 4 nM T47438 COHJ47 44435479 IC50 = 30 nM T47438 C0YU6V 44435480 IC50 = 10 nM T47438 C4KC1T 44435481 IC50 = 30 nM T47438 CFWA70 44435482 IC50 = 2.4 nM T47438 CD1H4G 44435483 IC50 = 26.1 nM T47438 C8DZ0C 44435484 IC50 = 30 nM T47438 CK95FN 44435485 IC50 = 2.2 nM T47438 CNXB96 44435486 IC50 = 1 nM T47438 C61BSW 44435487 IC50 < 34.6 nM T47438 CFLH45 44435488 IC50 = 64.8 nM T47438 C3VC7X 44435489 IC50 = 2.8 nM T47438 C8J2WB 44435490 IC50 = 141 nM T47438 CA9F6R 44435491 IC50 = 0.3 nM T47438 C4A5HJ 44435492 IC50 = 141 nM T47438 CCID56 44435493 IC50 = 12.9 nM T47438 CIO39Q 44435494 IC50 = 27.7 nM T47438 CX29JY 44435495 IC50 = 20.1 nM T47438 CXTH68 44435496 IC50 = 37.3 nM T47438 C32ZBN 44435497 IC50 = 16.8 nM T47438 C8ZU7E 44435530 IC50 = 13.6 nM T47438 CT6DY8 44438312 IC50 = 7.7 nM T47438 CJW0F5 44438313 IC50 = 26.8 nM T47438 C9YL5C 44438316 IC50 = 74.8 nM T47438 C4Q9NI 44438319 IC50 = 110 nM T47438 C6W2IH 44438321 IC50 = 152.5 nM T47438 C5GQ4C 44438322 IC50 = 164.5 nM T47438 CTYV56 44438323 IC50 = 0.7 nM T47438 C6Z9MA 44438324 IC50 = 5.3 nM T47438 CMJ73E 44438325 IC50 = 4.2 nM T47438 CU13SQ 44438327 IC50 = 7.9 nM T47438 C9B1UA 44438328 IC50 = 6.1 nM T47438 C97WJB 44438331 IC50 = 8.5 nM T47438 CET92A 44438332 IC50 = 15.4 nM T47438 CCQ4L2 44438334 IC50 = 3.7 nM T47438 C03BAR 44438335 IC50 = 4.5 nM T47438 C5S0ZB 44438337 IC50 = 5.5 nM T47438 CJW68H 44438338 IC50 = 9.7 nM T47438 C4A1IW 44438339 IC50 = 5.2 nM T47438 CR0WN3 44438340 IC50 = 3.6 nM T47438 CUTO72 44438341 IC50 = 120.4 nM T47438 C5PTA0 44438342 IC50 = 1.9 nM T47438 C2CYK4 44438343 IC50 = 2.1 nM T47438 C6AR1L 44438344 IC50 = 0.9 nM T47438 CH1A9C 44438345 IC50 = 0.3 nM T47438 CI9Z5D 44438347 IC50 = 16.8 nM T47438 CY4JS2 44438348 IC50 = 2.7 nM T47438 CQ1D4N 44438349 IC50 = 1.1 nM T47438 C5V0SU 44438350 IC50 = 2.4 nM T47438 CL5R1O 44438351 IC50 = 3.5 nM T47438 CVL65S 44438352 IC50 = 16.8 nM T47438 C7EV9J 44438385 IC50 = 172 nM T47438 C4QGK6 44438388 IC50 = 253 nM T47438 C5R0TJ 44438390 IC50 = 580 nM T47438 C7F6CI 44438393 IC50 = 440 nM T47438 CX8PM9 44438400 IC50 = 680 nM T47438 C1V4HC 44438402 IC50 = 629 nM T47438 CGAF37 44438404 IC50 = 290 nM T47438 CX0V5I 44438413 IC50 = 255 nM T47438 CW8R1G 44438417 IC50 = 219 nM T47438 CV98FE 44438419 IC50 = 217 nM T47438 C20UWR 44438421 IC50 > 1000 nM T47438 CTS16G 44438436 IC50 = 4.4 nM T47438 CFH2R8 44438651 IC50 = 13000 nM T47438 CLEM85 44438652 IC50 > 40000 nM T47438 C0JO3P 44438653 IC50 = 24000 nM T47438 C85LSF 44438654 IC50 = 38000 nM T47438 C0SWQ8 44438655 IC50 = 37000 nM T47438 CDHQ05 44438656 IC50 = 32000 nM T47438 CNQ7O0 44438657 IC50 = 13000 nM T47438 C5OS0L 44438658 IC50 > 40000 nM T47438 CCK6H4 44438659 IC50 = 16000 nM T47438 C3TEI7 44438660 IC50 = 19000 nM T47438 C73OXN 44438661 IC50 = 17000 nM T47438 CITL79 44438662 IC50 = 11000 nM T47438 CG9C3D 44440636 IC50 = 9 nM T47438 C7HY4S 44440637 IC50 = 6 nM T47438 CIPS34 44440638 IC50 = 8 nM T47438 C1RZ7M 44440639 IC50 = 59 nM T47438 C3XE9I 44440640 IC50 = 10 nM T47438 CN7H4Z 44440641 IC50 = 162 nM T47438 C7L8UV 44440642 IC50 = 43 nM T47438 CE7K6W 44440643 IC50 = 269 nM T47438 C1S3AI 44440644 IC50 = 3 nM T47438 CF1H9O 44440649 IC50 = 1 nM T47438 CJ5BS7 44440650 IC50 = 24 nM T47438 CH8P2F 44440651 IC50 = 1 nM T47438 C7WJL5 44440652 IC50 = 4 nM T47438 CK98ME 44440653 IC50 = 1.3 nM T47438 CN06BY 44440654 IC50 = 0.2 nM T47438 CSC65N 44440655 IC50 = 2 nM T47438 CY29QH 44440658 IC50 = 0.5 nM T47438 CV5T4N 44440666 IC50 = 2 nM T47438 CV3OC2 44440667 IC50 = 14 nM T47438 C7Z3TC 44440668 IC50 = 22 nM T47438 CRL40U 44440669 IC50 = 1.9 nM T47438 C29GPX 44440670 IC50 = 14 nM T47438 CTYP45 44440671 IC50 = 56 nM T47438 C9G1NJ 44440672 IC50 = 0.4 nM T47438 C86GRL 44440673 IC50 = 10 nM T47438 C0EM2O 44440674 IC50 = 750 nM T47438 CV6MS8 44441997 IC50 = 5.2 nM T47438 CDA0K3 44441998 IC50 = 18.5 nM T47438 C6VF9N 44441999 IC50 = 783 nM T47438 C5KPT0 44442000 IC50 > 1000 nM T47438 CSXU96 44442006 IC50 = 28.4 nM T47438 CF2NQ0 44442007 IC50 = 71.1 nM T47438 CX5V1C 44442008 IC50 = 103.5 nM T47438 C41NKY 44442009 IC50 > 1000 nM T47438 CH97AI 44442010 IC50 > 1000 nM T47438 C31THS 44442011 IC50 = 154.5 nM T47438 CPFY31 44442012 IC50 = 310.1 nM T47438 CWTI80 44442013 IC50 = 48.8 nM T47438 C4NST7 44442014 IC50 = 2.4 nM T47438 C3YR2W 44442017 IC50 = 8.1 nM T47438 C65KFB 44443276 EC50 = 10600 nM T47438 CFE6Y0 44443278 EC50 = 6200 nM T47438 CQLY72 44443990 IC50 = 3400 nM T47438 CI53PU 44443991 IC50 = 13 nM T47438 CB3O4E 44443992 IC50 = 3200 nM T47438 C7PEB3 44443993 IC50 = 9.7 nM T47438 CX96US 44443994 IC50 = 57 nM T47438 CU0A7X 44443995 IC50 = 9 nM T47438 CA2U1Z 44443997 IC50 = 830 nM T47438 CTX10R 44443998 IC50 = 7700 nM T47438 CL8VK6 44443999 IC50 = 180 nM T47438 C4V5PO 44444004 IC50 = 25 nM T47438 C7O1LX 44444015 IC50 = 21 nM T47438 CJD64U 44444017 IC50 = 65 nM T47438 CM95NK 44444020 IC50 = 13 nM T47438 C7ABX0 44444022 IC50 = 76 nM T47438 CKXE20 44444023 IC50 = 18 nM T47438 CXYJ51 44444048 IC50 = 45 nM T47438 CFAU69 44444049 IC50 = 33 nM T47438 CL18UT 44444050 IC50 = 12 nM T47438 CK2B9V 44444051 IC50 = 25 nM T47438 C3HGR6 44444054 IC50 = 41 nM T47438 C2UD9K 44444056 IC50 = 15 nM T47438 C63MJP 44444058 IC50 = 93 nM T47438 CED08T 44444059 IC50 = 29 nM T47438 CR43VX 44444063 IC50 = 64 nM T47438 C9BG8M 44444064 IC50 = 60 nM T47438 CC0Q9I 44444066 IC50 = 820 nM T47438 CM4FU3 44444067 IC50 = 660 nM T47438 CHTL58 44444068 IC50 = 130 nM T47438 CMXC12 44444069 IC50 = 550 nM T47438 CI8O7E 44444071 IC50 = 130 nM T47438 C49PGO 44444072 IC50 = 67 nM T47438 CLOY45 44444073 IC50 = 460 nM T47438 CL1HR0 44444074 IC50 = 120 nM T47438 C42NRC 44444075 IC50 = 340 nM T47438 CNI37J 44444077 IC50 = 27 nM T47438 C4CKQ7 44444078 IC50 = 690 nM T47438 C1YF2B 44444079 IC50 = 4500 nM T47438 C0YK9T 44444080 IC50 = 1400 nM T47438 C1DQN8 44444081 IC50 = 620 nM T47438 CDN8F5 44444082 IC50 = 110 nM T47438 CVG61I 44444083 IC50 = 85 nM T47438 CLP4E8 44444085 IC50 = 1100 nM T47438 CZ3O5X 44444087 IC50 = 67 nM T47438 C4J0ZO 44444088 IC50 = 470 nM T47438 CP0G8B 44444089 IC50 = 1000 nM T47438 CXD61J 44444090 IC50 = 330 nM T47438 C8TI3U 44444091 IC50 = 180 nM T47438 C7MTH4 44444092 IC50 = 150 nM T47438 CC2P1R 44444093 IC50 = 3900 nM T47438 C6CSF4 44444095 IC50 = 250 nM T47438 C1L2XV 44446139 IC50 = 5.1 nM T47438 CO57IE 44446141 IC50 = 7.3 nM T47438 CVOK90 44446142 IC50 = 13 nM T47438 C5T1SX 44446144 IC50 = 8.1 nM T47438 C0AEN8 44446145 IC50 = 6.9 nM T47438 CNGW15 44446147 IC50 = 14 nM T47438 CB52UA 44446149 IC50 = 15 nM T47438 C2G4DL 44446151 IC50 = 26 nM T47438 C3GDX0 44446153 IC50 = 1.6 nM T47438 C6G8RS 44446155 IC50 = 2.9 nM T47438 CO7Y2T 44446156 IC50 = 72 nM T47438 CEN64O 44446158 IC50 = 0.23 nM T47438 C0Q4XW 44446160 IC50 = 1.1 nM T47438 CMRT79 44446161 IC50 = 7.4 nM T47438 CWQ95D 44446163 IC50 = 288 nM T47438 C4S8ZQ 44446166 IC50 = 262 nM T47438 CZ3U6D 44446167 IC50 = 6.5 nM T47438 C2WQ3C 44446169 IC50 = 29 nM T47438 C71ELD 44446170 IC50 = 36 nM T47438 C6EK8F 44446171 IC50 = 50 nM T47438 C8ZK5B 44446172 IC50 = 3.1 nM T47438 C6PEY0 44446174 IC50 = 29 nM T47438 C5IW0Y 44446176 IC50 = 84 nM T47438 CMXW56 44446179 IC50 = 18 nM T47438 CNQH17 44446182 IC50 = 11 nM T47438 CK73CX 44446183 IC50 = 12 nM T47438 CPZA49 44446184 IC50 = 0.9 nM T47438 C4CZ9L 44446185 IC50 = 4.8 nM T47438 CW4Y9I 44446186 IC50 = 1.2 nM T47438 CIRM84 44446191 IC50 = 6.1 nM T47438 C5KCU2 44446192 IC50 = 61 nM T47438 CI69XS 44446193 IC50 = 0.75 nM T47438 CES2P4 44446194 IC50 = 15 nM T47438 C3MHK1 44446195 IC50 = 0.53 nM T47438 C7WKO1 44449123 IC50 = 8.7 nM T47438 CY27LD 44454961 IC50 > 10000 nM T47438 CK4BV0 44454962 IC50 = 257 nM T47438 CX5BZ2 44454988 IC50 > 10000 nM T47438 CD3QS7 44454989 IC50 = 685 nM T47438 C4BXT1 44455020 IC50 = 416 nM T47438 CT2UR5 44455050 IC50 = 212 nM T47438 CLQR53 44455051 IC50 = 105 nM T47438 CO01UH 44455052 IC50 = 81 nM T47438 CLRN39 44455054 IC50 = 62 nM T47438 CXYT35 44455355 IC50 = 23 nM T47438 CRWP10 44455388 IC50 > 10000 nM T47438 CJVC30 44455408 IC50 > 10000 nM T47438 C20GEX 44455409 IC50 > 10000 nM T47438 CO3V6X 44455431 IC50 > 10000 nM T47438 CYK50G 44455497 IC50 = 390 nM T47438 C4UK8G 44455523 IC50 = 3500 nM T47438 C8SFN2 44455525 IC50 = 2000 nM T47438 CNQ65C 44455577 IC50 = 150 nM T47438 CK75MF 44455580 IC50 = 17000 nM T47438 C8D6SZ 44455609 IC50 = 110 nM T47438 CPTW62 44455611 IC50 = 9000 nM T47438 CTW4Z5 44455643 IC50 = 150 nM T47438 C0O4PB 44455644 IC50 = 14000 nM T47438 C1C0OR 44455646 IC50 > 20000 nM T47438 CXYD92 44455729 IC50 = 30 nM T47438 C98DZW 44455731 IC50 = 8 nM T47438 CE4Q3W 44455732 IC50 = 2600 nM T47438 C2P5MJ 44455804 IC50 = 20 nM T47438 CQS0H9 44455828 IC50 > 20000 nM T47438 C85CZH 44571533 IC50 = 0.7 nM T47438 C24IJZ 44571534 IC50 = 0.6 nM T47438 CT0Z2K 44626366 IC50 > 50000 nM T47438 CI1G4L 44814464 IC50 = 13000 nM T47438 CJG7H3 44815008 IC50 = 22000 nM T47438 CGEF05 45101437 IC50 = 0.67 nM T47438 CW5DH0 45263545 IC50 = 3 nM T47438 CZP0C2 45263546 IC50 = 83 nM T47438 CFA23Y 45263651 IC50 = 0.8 nM T47438 C79OBA 45263654 IC50 = 7.9 nM T47438 C19VMP 45279238 IC50 = 0.75 nM T47438 CAI2S3 45279243 IC50 = 4 nM T47438 CVE8H0 45279329 IC50 = 32 nM T47438 CMU1Y2 45279330 IC50 = 20 nM T47438 C98ZUP 45279331 IC50 = 175 nM T47438 CNL75F 45279417 IC50 = 94 nM T47438 CO4ZS2 45279505 IC50 = 26 nM T47438 CY3H1B 45279506 IC50 = 1 nM T47438 CVE91H 45279510 IC50 = 10 nM T47438 C1IT0C 45279600 IC50 = 2229 nM T47438 CXU8W7 45485422 IC50 = 2.9 nM T47438 C64YKE 45485436 IC50 = 4.2 nM T47438 C8Q0FP 45485446 IC50 = 3.2 nM T47438 CG2JD6 45485450 IC50 = 0.31 nM T47438 CM3DO4 45485456 IC50 = 0.37 nM T47438 CAO31T 45485464 IC50 = 0.41 nM T47438 C8JES7 45485471 IC50 = 0.58 nM T47438 C5UBN2 45485490 IC50 = 1.5 nM T47438 CZU9L2 45485491 IC50 = 0.2 nM T47438 CK6ZT7 45485492 IC50 = 0.62 nM T47438 CJ6TP3 45485495 IC50 = 0.26 nM T47438 CR2FZ0 45485496 IC50 = 0.44 nM T47438 CEWX31 45485523 IC50 = 0.17 nM T47438 COU45W 45485527 IC50 = 0.26 nM T47438 CV9W4F 45485533 IC50 = 0.26 nM T47438 CIWV94 45485553 IC50 = 0.24 nM T47438 CDZ84U 45487083 IC50 = 2510 nM T47438 CP7O3K 45487084 IC50 = 4889 nM T47438 CMH59T 45487090 IC50 = 5722 nM T47438 CN86WT 45487093 IC50 = 0.52 nM T47438 CK8J0C 45487094 IC50 = 66 nM T47438 C9WD4X 45487096 IC50 = 202 nM T47438 C6Q5MP 45487102 IC50 = 678 nM T47438 CS20OB 45487103 IC50 = 1109 nM T47438 C29SDN 45487104 IC50 = 70 nM T47438 C5EO7Y 45487109 IC50 = 989 nM T47438 CA8BF4 45487115 IC50 = 8813 nM T47438 CU90YF 45487122 IC50 = 9 nM T47438 CH0N3P 45487123 IC50 = 194 nM T47438 C4EU3H 45487124 IC50 = 2 nM T47438 CAP86G 45487130 IC50 = 1066 nM T47438 C5RJ4D 45487131 IC50 = 826 nM T47438 CGVJ06 45487146 IC50 = 1 nM T47438 CGUL09 45487151 IC50 = 5654 nM T47438 CUC2W8 46186977 EC50 = 47600 nM T47438 CE9U3O 46189877 IC50 = 13300 nM T47438 CN8C1E 46200343 IC50 = 191 nM T47438 C92RAS 46200344 IC50 = 72 nM T47438 CDK02H 46201982 IC50 = 230 nM T47438 CRLM46 46201983 IC50 = 33 nM T47438 CXAK48 46203600 IC50 = 300 nM T47438 C40JBU 46203602 IC50 = 76 nM T47438 CMG2U0 46204901 IC50 = 87 nM T47438 CTXE90 46205227 IC50 = 37 nM T47438 C6UNV9 46205555 IC50 = 56 nM T47438 CLG92T 46205556 IC50 = 5400 nM T47438 CK1ZG6 46205872 IC50 = 44 nM T47438 C8ONI5 46205873 IC50 = 1900 nM T47438 CFO2S8 46205876 IC50 = 19000 nM T47438 CS7A1F 46206542 IC50 = 530 nM T47438 C64UTP 46206544 IC50 = 3100 nM T47438 CVW24X 46206545 IC50 = 80 nM T47438 CN7QE6 46206546 IC50 = 100 nM T47438 C4K3DZ 46206874 IC50 = 3300 nM T47438 CJ79UT 46206875 IC50 = 120 nM T47438 CYP2H6 46206879 IC50 = 820 nM T47438 CK4TI1 46214177 IC50 = 130 nM T47438 CE02DJ 46214505 IC50 = 1260 nM T47438 CQ5G0O 46214506 IC50 = 37 nM T47438 CQ1Z0D 46214507 IC50 = 140 nM T47438 CPF0J9 46214673 IC50 = 39 nM T47438 CV2Q4F 46214674 IC50 = 49 nM T47438 CEB7L5 46214832 IC50 = 35 nM T47438 C8KE9V 46214983 IC50 = 2500 nM T47438 C5TEA2 46214986 IC50 = 1100 nM T47438 CME1P7 46215156 IC50 = 24 nM T47438 CX5BE1 46215326 IC50 = 16 nM T47438 CL58QM 46215511 IC50 = 40 nM T47438 C0QS3H 46215512 IC50 = 95 nM T47438 C35ZCM 46215514 IC50 = 240 nM T47438 C5DV7T 46216355 IC50 = 41 nM T47438 CT6J2S 46216529 IC50 = 41 nM T47438 CL86HB 46216678 EC50 = 501.19 nM T47438 CX7K3M 46216736 IC50 = 6140 nM T47438 C83ZQU 46225338 IC50 > 10000 nM T47438 CN74XF 46225339 IC50 = 390 nM T47438 C43PME 46225360 IC50 = 600 nM T47438 C12LPT 46225361 IC50 = 640 nM T47438 C8A3DL 46228934 IC50 > 30000 nM T47438 CR4KT7 46229901 IC50 > 50000 nM T47438 CW4P2I 46229902 IC50 > 50000 nM T47438 C5FB9H 46229972 IC50 > 50000 nM T47438 C9L8MQ 46229973 IC50 > 50000 nM T47438 CJAH09 46229974 IC50 = 34430 nM T47438 COFP27 46231466 IC50 = 1995.26 nM T47438 CD7CJ3 46231467 IC50 = 10000 nM T47438 C86UDB 46231469 EC50 = 10000 nM T47438 CPJ4R8 46231471 IC50 = 1000 nM T47438 C19JAS 46231522 IC50 = 630.96 nM T47438 CMF8X1 46231524 IC50 = 630.96 nM T47438 CFAK81 46231526 IC50 = 251.19 nM T47438 C1G9YE 46231528 IC50 = 1258.93 nM T47438 CP9Y1S 46231577 EC50 = 501.19 nM T47438 CS2EI9 46231579 IC50 = 10000 nM T47438 C4U6HW 46231628 IC50 = 25118.86 nM T47438 CNH5D1 46231630 IC50 = 1258.93 nM T47438 CC03FA 46231632 IC50 = 1584.89 nM T47438 C7XNM1 46231634 IC50 = 1995.26 nM T47438 CUPG59 46231688 IC50 = 316.23 nM T47438 C2GIB6 46231690 IC50 = 1258.93 nM T47438 COA9P3 46231692 IC50 = 398.11 nM T47438 C5H0AL 46231694 IC50 = 794.33 nM T47438 CZ36XF 46231747 IC50 = 398.11 nM T47438 CSA40G 46231749 IC50 = 794.33 nM T47438 CH0CA1 46231751 IC50 = 1258.93 nM T47438 C0XBY7 46231753 IC50 = 630.96 nM T47438 CDA42Z 46231821 IC50 = 12589.25 nM T47438 CKT0W9 46236732 IC50 = 0.35 nM T47438 CP4L1C 46236733 IC50 = 250 nM T47438 CO0QT7 46841575 IC50 = 26 nM T47438 CO31WX 46861576 IC50 = 16 nM T47438 C8EX6T 46864718 EC50 = 6 nM T47438 CT5A7F 46871758 IC50 = 54 nM T47438 CIS65O 46871825 IC50 = 1.9 nM T47438 C5Y2ZB 46878651 EC50 = 1400 nM T47438 C3UO4V 46878691 EC50 = 9300 nM T47438 CBEO79 46878692 EC50 = 12600 nM T47438 C3JCD4 46878693 EC50 = 9200 nM T47438 CH3Y9O 46878694 EC50 > 40000 nM T47438 CUK40A 46878737 EC50 = 7600 nM T47438 C2Z9UW 46878738 EC50 > 80000 nM T47438 CWA51E 46878739 EC50 > 80000 nM T47438 C41OTL 46878740 EC50 = 16100 nM T47438 CT1N2L 46878785 EC50 > 40000 nM T47438 CI23FY 46878786 IC50 = 36100 nM T47438 CS6N2R 46878787 EC50 > 40000 nM T47438 CEN9Y3 46878788 EC50 > 40000 nM T47438 CR1ZX3 46878848 EC50 > 80000 nM T47438 CFRJ50 46878849 EC50 > 80000 nM T47438 C5WXJ0 46878850 EC50 > 40000 nM T47438 CC29YQ 46878851 EC50 > 40000 nM T47438 C9GAN2 46878852 EC50 = 47600 nM T47438 C7VA3G 46883541 IC50 = 2.1 nM T47438 CRAO48 46883741 IC50 = 5000 nM T47438 CFI6X4 46883745 IC50 = 20 nM T47438 C3DSI2 46883776 IC50 = 651 nM T47438 CP8Q6Y 46883777 IC50 = 467 nM T47438 CCPX03 46883778 IC50 = 6 nM T47438 COZ41D 46883779 IC50 = 1 nM T47438 C8S7FD 46883804 IC50 = 0.77 nM T47438 CF82LP 46884323 IC50 = 1698 nM T47438 CD50RE 46884324 IC50 = 760 nM T47438 CEW94S 46884370 IC50 = 662 nM T47438 C2YZ8W 46884456 IC50 = 557 nM T47438 CNH6Y3 46884457 IC50 = 1.01 nM T47438 CA67FX 46884483 IC50 = 3.7 nM T47438 CY0G3Q 46884484 IC50 = 22.4 nM T47438 CB7MI5 46884678 IC50 = 9200 nM T47438 COW3L9 46884679 IC50 > 50000 nM T47438 CM78KJ 46884705 IC50 > 50000 nM T47438 CJG0C1 46884792 IC50 = 9100 nM T47438 C1MP7S 46890758 IC50 = 25072 nM T47438 CEW8I9 46890759 IC50 = 187 nM T47438 CT5KD7 46890760 IC50 = 71 nM T47438 C6UBC0 46890761 IC50 = 574 nM T47438 CU20TA 46890816 IC50 = 418 nM T47438 C40CHX 46890817 IC50 = 358 nM T47438 CX9KP3 46890818 IC50 = 771 nM T47438 C9HBP7 46890819 IC50 = 304 nM T47438 CI6SX2 46890820 IC50 = 403 nM T47438 C8YU2V 46890880 IC50 = 304 nM T47438 CY6BV2 46890881 IC50 = 138 nM T47438 C5J8IW 46890882 IC50 = 34 nM T47438 C6CXV3 46890883 IC50 = 13 nM T47438 CKW2T8 46890943 IC50 = 2656 nM T47438 CCH1L9 46890944 IC50 = 995 nM T47438 CXO39V 46890945 IC50 = 235 nM T47438 C9LPA4 46891002 IC50 = 6209 nM T47438 CL47FR 46891003 IC50 = 576 nM T47438 C4VWG2 46891052 IC50 = 25 nM T47438 CMGW50 46891411 IC50 = 546 nM T47438 C6EA2X 46891412 IC50 = 288 nM T47438 CRBX43 46891413 IC50 > 40000 nM T47438 C24XZM 46891455 IC50 > 40000 nM T47438 CRAM45 46891456 IC50 > 40000 nM T47438 CNAX47 46891457 IC50 > 40000 nM T47438 CBL1E2 46891458 IC50 > 40000 nM T47438 CN4RS8 46891517 IC50 = 2302 nM T47438 C2C3LG 46891518 IC50 = 2792 nM T47438 C9R5UL 46891519 IC50 > 40000 nM T47438 CF12WN 46891520 IC50 > 40000 nM T47438 C1B8DK 46891521 IC50 = 18334 nM T47438 C15OSQ 46891575 IC50 > 40000 nM T47438 CLO7S1 46891576 IC50 > 40000 nM T47438 C61NMK 46891577 IC50 = 4000 nM T47438 CZ8V9I 46891578 IC50 = 2361 nM T47438 C4KNU1 46891579 IC50 = 6704 nM T47438 CZ7C1J 46893145 IC50 = 130 nM T47438 CP2FI0 46912223 IC50 = 1.7 nM T47438 CF35QN 49865652 IC50 = 3502 nM T47438 CYNH04 49865736 IC50 = 229 nM T47438 CW2M9C 49865787 IC50 = 7100 nM T47438 CD49WA 49865788 IC50 = 106 nM T47438 C79LFV 49865865 IC50 = 85 nM T47438 C3J7YR 49865866 IC50 = 503 nM T47438 CWX5Y7 49865867 IC50 = 73 nM T47438 CED86P 49865925 IC50 > 20000 nM T47438 CL3K5Q 49865926 IC50 > 20 nM T47438 C4Z0BG 49866251 IC50 = 163 nM T47438 C7GR0H 49872381 IC50 = 40 nM T47438 CD1X3U 49872384 IC50 = 28 nM T47438 C6B0NT 49872385 IC50 = 60 nM T47438 CZML42 49872482 IC50 = 68 nM T47438 C60RMP 49872483 IC50 = 19 nM T47438 CA3QJ9 50898349 IC50 = 122 nM T47438 CZIS04 50899302 IC50 = 900 nM T47438 C4BD6H 52935148 IC50 = 158 nM T47438 C3Q6TV 52939724 IC50 = 200 nM T47438 CF86AB 52946557 IC50 = 800 nM T47438 CBS28G 52947827 IC50 = 1400 nM T47438 CTV15R 52949026 IC50 = 1500 nM T47438 CWQ8Y2 53307787 IC50 = 300 nM T47438 CR7TD8 53307788 IC50 = 200 nM T47438 C8XR3L 53316726 IC50 = 342 nM T47438 CVY45A 53316727 IC50 = 19316 nM T47438 C1SBC9 53316728 IC50 = 1919 nM T47438 CR3E5C 53316729 IC50 = 448 nM T47438 CU72TL 53316730 IC50 = 164 nM T47438 C9RK8W 53317504 IC50 = 1860 nM T47438 CXT58Z 53318019 IC50 = 20000 nM T47438 C37ZAQ 53318697 IC50 = 370 nM T47438 CBLD50 53318698 IC50 = 200 nM T47438 CIN82X 53319361 IC50 = 537 nM T47438 C68CRW 53319362 IC50 = 356 nM T47438 C5YZC0 53319363 IC50 = 440 nM T47438 C8U2PO 53319364 IC50 = 875 nM T47438 CC37JA 53319365 IC50 = 935 nM T47438 CM4H0Y 53319366 IC50 = 209 nM T47438 CUG7V3 53320013 IC50 = 2080 nM T47438 CS04NZ 53320014 IC50 = 1070 nM T47438 CKJQ81 53320673 IC50 = 156 nM T47438 C0SU6P 53320674 IC50 = 2531 nM T47438 CMG8J3 53320675 IC50 = 1409 nM T47438 CQD62W 53321323 IC50 = 540 nM T47438 COT69M 53321324 IC50 = 320 nM T47438 CJO8K6 53321365 IC50 = 1406 nM T47438 C92ZPY 53321966 IC50 = 126 nM T47438 CUP16W 53321967 IC50 = 1392 nM T47438 C4O6RY 53323317 IC50 = 145 nM T47438 CJT3O4 53323318 IC50 = 16374 nM T47438 CT0IN8 53323319 IC50 = 485 nM T47438 CMG85A 53323320 IC50 = 465 nM T47438 C5RDB1 53323321 IC50 = 540 nM T47438 C8ZHY7 53323979 IC50 > 10000 nM T47438 C9Q1ND 53324647 IC50 = 20000 nM T47438 CV9XG0 53324648 IC50 = 2069 nM T47438 CB35NA 53324649 IC50 = 2215 nM T47438 C2FV4W 53324650 IC50 = 201 nM T47438 CUO1R8 53325274 IC50 = 1290 nM T47438 CZB7M2 53325275 IC50 = 1690 nM T47438 CLV49B 53325838 IC50 = 649 nM T47438 C7GQK5 53325949 IC50 = 552 nM T47438 C3KWC5 53326627 IC50 = 1650 nM T47438 CZ8DU9 53326926 IC50 = 619 nM T47438 CF67UL 53327840 IC50 = 0.4 nM T47438 C6ACY1 53466872 IC50 > 4000 nM T47438 C4U5IX 53493001 EC50 = 70 nM T47438 CMNA20 54580854 IC50 = 2.7 nM T47438 C46ZWI 54580879 IC50 = 1.7 nM T47438 CD45JK 54581914 IC50 = 263 nM T47438 C6EPJ0 54581915 IC50 = 82.8 nM T47438 CTCM02 54581934 IC50 = 226 nM T47438 C50EXN 54581935 IC50 = 0.8 nM T47438 C5RDG6 54581936 IC50 > 10000 nM T47438 CJ1WZ3 54582829 IC50 = 52.7 nM T47438 C94LQC 54582858 IC50 = 7.8 nM T47438 C3QVP4 54582859 IC50 = 9.4 nM T47438 CRAW75 54582860 IC50 = 3100 nM T47438 CHX16Y 54582861 IC50 = 250 nM T47438 CIKC16 54582862 IC50 = 480 nM T47438 CZ4DV0 54582863 IC50 = 8.9 nM T47438 CY81FK 54582864 IC50 = 5.4 nM T47438 CUL04M 54583866 IC50 = 21.6 nM T47438 CA3UH9 54583867 IC50 = 31 nM T47438 C0O8UB 54583868 IC50 = 2.9 nM T47438 CIT94F 54583869 IC50 = 3.3 nM T47438 CFO6L2 54583870 IC50 = 4.6 nM T47438 CFL7C6 54584820 IC50 = 2.5 nM T47438 CTO6N3 54584821 IC50 = 148 nM T47438 CZ5IA1 54585612 IC50 = 3.8 nM T47438 CZR3A2 54585748 IC50 = 0.39 nM T47438 CQH3O5 54585770 IC50 = 64.6 nM T47438 C0W3NV 54585771 IC50 = 310 nM T47438 CM45DH 54585772 IC50 = 19.5 nM T47438 CJM86T 54585773 IC50 = 19.3 nM T47438 CM6KH7 54585774 IC50 = 6.9 nM T47438 CCK9Z3 54586727 IC50 = 14.6 nM T47438 C8TMD3 54586758 IC50 = 3.6 nM T47438 C2G0RU 54586759 IC50 = 4.3 nM T47438 CV1L4K 54586760 IC50 = 8.2 nM T47438 C6L0WH 54586761 IC50 = 4.9 nM T47438 CYT89D 54587765 IC50 = 1.2 nM T47438 CE19HM 54587781 IC50 = 0.4 nM T47438 C5GC3J 54587782 IC50 = 45.7 nM T47438 C8NYA1 54587783 IC50 = 7.9 nM T47438 C0AIO8 54587784 IC50 = 53.9 nM T47438 CNA7I0 54587785 IC50 = 93.3 nM T47438 C0VYX8 54669875 IC50 = 7.99 nM T47438 C24UKQ 54764004 IC50 = 125.89 nM T47438 C9LF2N 56592447 EC50 = 30 nM T47438 CQ1GO6 56658871 IC50 = 10457 nM T47438 CE05WK 56658872 IC50 = 8 nM T47438 CTKA80 56659252 EC50 = 21000 nM T47438 CI48MU 56659253 EC50 = 19000 nM T47438 C3TAV6 56659254 EC50 = 49000 nM T47438 C4KGE6 56659627 IC50 = 794.33 nM T47438 CXZW56 56659628 IC50 > 100000 nM T47438 CS4N2M 56659870 IC50 = 1640 nM T47438 CI1Z4B 56659871 IC50 = 1000 nM T47438 C0PSG1 56659872 IC50 = 270 nM T47438 C2RX1T 56662356 IC50 = 187 nM T47438 CWS15Q 56662733 IC50 = 12900 nM T47438 CU25CK 56662734 IC50 = 89000 nM T47438 CXSD38 56663088 IC50 = 316.23 nM T47438 CB9ZN5 56663089 IC50 = 50118.72 nM T47438 C1IPX6 56663090 IC50 = 1995.26 nM T47438 CN70JC 56663117 IC50 = 316.23 nM T47438 CK5FY6 56663118 IC50 = 100 nM T47438 CXE41B 56663331 IC50 = 7060 nM T47438 C0PTB8 56663332 IC50 = 7010 nM T47438 CU6NX4 56665650 IC50 = 29 nM T47438 CV04XS 56666134 IC50 > 500 nM T47438 CJ8AQ3 56666135 IC50 > 80000 nM T47438 CZE94O 56666199 IC50 = 32000 nM T47438 C01YFA 56666200 IC50 > 80000 nM T47438 C9SC6L 56666757 IC50 = 5710 nM T47438 C4MFS5 56666758 IC50 = 450 nM T47438 CF0KZ2 56666759 IC50 = 820 nM T47438 C62JDU 56666760 IC50 = 410 nM T47438 C1GH7Y 56669242 IC50 = 18719 nM T47438 C1P6WA 56669243 IC50 = 29 nM T47438 CK71EP 56669244 IC50 = 888 nM T47438 C5D7ZT 56669536 EC50 = 12000 nM T47438 C2F4UM 56669537 EC50 = 8000 nM T47438 CA1ME9 56669597 IC50 = 80000 nM T47438 CP8M7G 56669598 IC50 = 27000 nM T47438 C25AQX 56669599 IC50 > 80000 nM T47438 C3L4ZK 56669956 IC50 = 10000 nM T47438 C06PUJ 56669957 IC50 = 501.19 nM T47438 C3U4AP 56669979 IC50 = 79.43 nM T47438 C78SDI 56669980 IC50 = 158.49 nM T47438 CZO49F 56670192 IC50 = 2640 nM T47438 CJ8P3S 56672571 IC50 = 21 nM T47438 C3GV1C 56672708 IC50 = 4 nM T47438 CTD9Z3 56672709 IC50 = 4 nM T47438 C8WG2N 56672710 IC50 = 767 nM T47438 CNR2P1 56673049 EC50 = 21000 nM T47438 C7C4VZ 56673050 EC50 = 32000 nM T47438 CPUK68 56673051 EC50 > 80000 nM T47438 CS7KW0 56673052 IC50 > 80000 nM T47438 CCQK10 56673053 IC50 = 102000 nM T47438 CZPU76 56673054 EC50 > 40000 nM T47438 CE78CJ 56673118 IC50 = 104000 nM T47438 CI8P9J 56673119 EC50 = 15000 nM T47438 CXM90K 56673464 IC50 = 6309.57 nM T47438 C2GN9F 56673465 IC50 = 3162.28 nM T47438 CL0Q3N 56673466 IC50 = 398.11 nM T47438 C7E3IP 56673494 IC50 = 100 nM T47438 CL4P9H 56673495 IC50 = 50.12 nM T47438 C4G0YE 56673715 IC50 = 1220 nM T47438 CWZV47 56673716 IC50 = 220 nM T47438 C1KW9Z 56673717 IC50 = 4040 nM T47438 CJUC47 56676069 IC50 = 7 nM T47438 CQV4B5 56676365 IC50 = 105000 nM T47438 CN81GL 56676366 EC50 = 21000 nM T47438 C9YV7U 56676367 EC50 > 10000 nM T47438 C6DAW2 56676435 IC50 = 31000 nM T47438 C6KCR5 56676736 IC50 = 79.43 nM T47438 C70DIW 56676779 IC50 = 199.53 nM T47438 C4KL0A 56676780 IC50 = 5011.87 nM T47438 C79ILY 56677020 IC50 = 1940 nM T47438 CL7AW3 56677021 IC50 = 780 nM T47438 CVXN71 56679251 IC50 = 14 nM T47438 CUHO31 56679252 IC50 = 16 nM T47438 C82YOE 56679400 IC50 = 28 nM T47438 C0C3TN 56679401 IC50 = 437 nM T47438 C7YM2G 56679402 IC50 = 149 nM T47438 C7QRM2 56679701 EC50 = 50000 nM T47438 CZO95E 56679702 IC50 = 24000 nM T47438 C4VU6Z 56679703 IC50 > 40000 nM T47438 C4LO5Q 56679704 IC50 > 80000 nM T47438 CQ8K7M 56680096 IC50 = 398.11 nM T47438 C6EO3N 56680128 IC50 = 39.81 nM T47438 C2KEV0 56680350 IC50 > 10000 nM T47438 C9DTH0 56680351 IC50 = 490 nM T47438 CMR0J9 56680352 IC50 = 1410 nM T47438 CDXT81 56681654 IC50 = 270 nM T47438 CYZ34G 56682694 IC50 = 22 nM T47438 C13LZJ 56683026 EC50 = 23000 nM T47438 CTC48A 56683027 EC50 > 80000 nM T47438 CVR0H1 56683437 IC50 = 251.19 nM T47438 CR8N0J 56683438 IC50 = 10000 nM T47438 C24XYT 56683439 IC50 = 251.19 nM T47438 C2MJ4D 56683476 IC50 = 2511.89 nM T47438 CKF29M 56683680 IC50 > 10000 nM T47438 C4X7IP 56683681 IC50 = 1440 nM T47438 C18ADK 56833940 IC50 = 16.9 nM T47438 C1MFZ4 56833941 IC50 = 16.5 nM T47438 C3I9PO 56833942 IC50 = 72.4 nM T47438 CHC9A6 56833943 IC50 = 49 nM T47438 CD30YZ 56833944 IC50 = 49.5 nM T47438 CO3EV9 56833945 IC50 = 12.3 nM T47438 CT16AO 56834043 IC50 = 16.6 nM T47438 CMI5T6 56834044 IC50 = 11.7 nM T47438 CCNF23 56834045 IC50 = 7.97 nM T47438 CMOU39 56834046 IC50 = 27.9 nM T47438 C4LQM9 56834047 IC50 = 33.8 nM T47438 CCP0K8 56834048 IC50 = 45.2 nM T47438 CP0VQ2 56834146 IC50 = 8.58 nM T47438 CMPT46 56834147 IC50 = 5.25 nM T47438 CD0K6U 56834148 IC50 = 7.53 nM T47438 CTDB01 56834149 IC50 = 13.4 nM T47438 CK4RN1 56834150 IC50 = 11.2 nM T47438 CP82BX 56834151 IC50 = 5.51 nM T47438 C6I8SK 56834259 IC50 = 44.5 nM T47438 CSCR53 56834260 IC50 = 16.4 nM T47438 CO6L5V 56834261 IC50 = 10.8 nM T47438 CJY10S 56834262 IC50 = 6.46 nM T47438 CQ84ZA 56945122 EC50 = 29 nM T47438 C0WBY6 56945991 IC50 = 187 nM T47438 C87GZI 56946207 IC50 = 122 nM T47438 C6A2FU 56946208 IC50 = 18833 nM T47438 CMAU62 56946312 IC50 = 80 nM T47438 C2E5TO 56946313 IC50 = 199 nM T47438 CHRU78 56946423 IC50 = 29 nM T47438 CQB9G8 56946424 IC50 = 7643 nM T47438 CI28DU 56946526 IC50 = 16237 nM T47438 C4MDZ6 56946527 IC50 = 89 nM T47438 C1KI4X 56946528 IC50 = 3210 nM T47438 C52OXA 56946529 IC50 = 26 nM T47438 CKM18B 56946627 IC50 = 53 nM T47438 CQ2MT0 56946628 IC50 = 117 nM T47438 CDQN37 56946629 IC50 = 21 nM T47438 C5VIB3 56946630 IC50 = 103 nM T47438 CSE28N 56946631 IC50 = 106 nM T47438 CE68HR 56953105 IC50 = 1.77 nM T47438 CJ3O9S 57327010 IC50 = 0.27 nM T47438 CYCP25 57327180 IC50 = 0.178 nM T47438 C30IZU 57384527 IC50 = 0.99 nM T47438 CQA35K 57384528 IC50 = 22.5 nM T47438 CJ3C9M 57384790 IC50 = 87.1 nM T47438 CGL94D 57384791 IC50 = 11.1 nM T47438 CMJ10O 57384792 IC50 = 6.92 nM T47438 C3MP2C 57384793 IC50 = 14.7 nM T47438 C0X1DZ 57384794 IC50 = 4.77 nM T47438 CN0YS7 57385030 IC50 = 7.47 nM T47438 CF5D1K 57385031 IC50 = 9.6 nM T47438 CEH5V4 57385032 IC50 = 4.11 nM T47438 C9LM2N 57385033 IC50 = 24.4 nM T47438 CSA8N6 57385034 IC50 = 12.1 nM T47438 CWZY54 57385280 IC50 = 45.5 nM T47438 CRO35Q 57385281 IC50 = 12.3 nM T47438 CMDX46 57390296 IC50 > 1250 nM T47438 C97PNB 57390896 IC50 = 56 nM T47438 CL2C3I 57392070 IC50 = 52 nM T47438 CX7L1C 57392134 IC50 = 2868 nM T47438 CRXD10 57392696 IC50 = 60 nM T47438 C5IM8F 57393826 IC50 = 3431 nM T47438 CHET54 57393827 IC50 = 3358 nM T47438 CJIZ48 57397373 IC50 = 999 nM T47438 CH32BO 57397434 IC50 > 5000 nM T47438 CO14BW 57397444 IC50 = 376 nM T47438 CVRD17 57399109 IC50 > 40000 nM T47438 CZLD01 57399119 IC50 = 5548 nM T47438 CW2DO9 57399120 IC50 = 483 nM T47438 CG7NW9 57400793 IC50 = 675 nM T47438 CR6AE3 57400851 EC50 = 1500 nM T47438 CYVN84 57402550 IC50 = 733 nM T47438 C5XF1Z 57402551 IC50 = 86 nM T47438 CSCH73 57404337 IC50 > 50000 nM T47438 C4QT2R 57404351 IC50 = 1000 nM T47438 CS1V8U 57404352 IC50 = 4 nM T47438 CKU6E8 57404500 IC50 > 50000 nM T47438 CXHN06 57987388 IC50 = 120 nM T47438 CXW7P5 58063504 IC50 = 18 nM T47438 C1XI2O 58063517 IC50 = 145 nM T47438 CEWR70 58065681 IC50 = 183 nM T47438 C15MAW 58065745 IC50 = 17 nM T47438 CRZH72 58173522 IC50 = 120 nM T47438 CGTB71 58445369 IC50 = 250 nM T47438 C0IZ4O 58469132 IC50 > 20000 nM T47438 CE94VP 58528692 IC50 = 210 nM T47438 CR4GK2 58528697 IC50 = 83 nM T47438 C1JO3I 58528715 IC50 = 9000 nM T47438 CH83XK 58528726 IC50 = 250 nM T47438 C5R7ZG 58528729 IC50 = 130 nM T47438 CS8WO1 58528732 IC50 = 39 nM T47438 CX3SQ7 58528738 IC50 = 88 nM T47438 CZEK86 58528741 IC50 = 140 nM T47438 C0VL2K 58528743 IC50 = 1500 nM T47438 CU2G9R 58528758 IC50 = 73 nM T47438 CY9SH8 58528759 IC50 = 400 nM T47438 C54KGY 58528775 IC50 = 580 nM T47438 C70BOM 58528779 IC50 = 3700 nM T47438 CLE51O 58528784 IC50 = 6700 nM T47438 C6P8SD 58548876 IC50 = 52 nM T47438 C0N5GT 58850279 IC50 = 4 nM T47438 C83YXM 58910631 IC50 = 130 nM T47438 CP91WC 58910757 EC50 = 1500 nM T47438 CG3Y5M 58950709 IC50 = 6.8 nM T47438 CVBT13 59201219 IC50 = 45 nM T47438 C1E3XT 59472470 IC50 = 42 nM T47438 C92NPY 59472493 IC50 = 1250 nM T47438 CL4F1U 59472507 IC50 = 8710 nM T47438 CG1ZH6 59472511 IC50 = 3980 nM T47438 CHU2S4 59472516 IC50 = 200 nM T47438 CW4I0H 59472517 IC50 = 40 nM T47438 C4RZ7E 59472522 IC50 = 390 nM T47438 CKS31U 59472524 IC50 = 180 nM T47438 C35EKB 59472530 IC50 = 10 nM T47438 CLB40A 59472544 IC50 = 78 nM T47438 CL9Y0P 59472546 IC50 = 680 nM T47438 CXH19J 59472574 IC50 = 30 nM T47438 C51KUS 59472588 IC50 = 70 nM T47438 CPH07V 59472599 IC50 = 78 nM T47438 CS87XI 59472603 IC50 = 150 nM T47438 CI8H4T 59472630 IC50 = 1630 nM T47438 CXO21N 59472637 IC50 = 3860 nM T47438 CH0S6A 59472641 IC50 = 430 nM T47438 C0LBN5 59472644 IC50 = 4850 nM T47438 C4SR9V 59472646 IC50 = 1270 nM T47438 C6D7LS 59472679 IC50 = 160 nM T47438 C8UMR6 59472684 IC50 = 40 nM T47438 C1ME7D 59472698 IC50 = 2010 nM T47438 CYO06N 59472699 IC50 = 370 nM T47438 C6XDH2 59472707 IC50 = 90 nM T47438 CF72WU 59472713 IC50 = 440 nM T47438 C9L0GJ 59472717 IC50 = 4420 nM T47438 CGD8W0 59472725 IC50 = 38 nM T47438 C2T4EU 59472735 IC50 = 380 nM T47438 CJR3K7 59472756 IC50 = 180 nM T47438 C1RUN6 59472765 IC50 = 70 nM T47438 CZ52KP 59472771 IC50 = 940 nM T47438 CB3X0F 59472773 IC50 = 1080 nM T47438 C6YZR8 59472775 IC50 = 480 nM T47438 CDOV85 59472789 IC50 = 1110 nM T47438 CWD0K3 59472815 IC50 = 270 nM T47438 C05YQD 59472822 IC50 = 28 nM T47438 C15JGP 59472849 IC50 = 1190 nM T47438 CM0G7S 59472858 IC50 = 940 nM T47438 CEP94I 59472861 IC50 = 80 nM T47438 CLH47W 59472872 IC50 = 150 nM T47438 CKGD30 59570713 IC50 > 100000 nM T47438 C18TXZ 60150510 IC50 = 10 nM T47438 C30UIB 60150707 IC50 = 9 nM T47438 C3V4UC 66549618 IC50 > 5000 nM T47438 CM4QT6 66551384 IC50 = 18 nM T47438 CO27HW 66551578 IC50 = 17 nM T47438 CZX69Y 66551579 IC50 = 25 nM T47438 CY7XR2 66551580 IC50 = 59 nM T47438 CPGZ81 66551772 IC50 = 30 nM T47438 CSP8G3 66678794 IC50 = 145 nM T47438 C9VW4M 66679082 IC50 = 25 nM T47438 CF6X2S 66679323 IC50 = 43 nM T47438 CK1J6R 66679335 IC50 = 69 nM T47438 C96BLD 66679340 IC50 = 5289 nM T47438 C79GQM 66679372 IC50 = 107 nM T47438 C8LMK0 66679376 IC50 = 2113 nM T47438 CZKV14 66679405 IC50 = 17 nM T47438 CYEL45 66679447 IC50 = 82 nM T47438 C1CUA9 66679503 IC50 = 696 nM T47438 CJ0KL5 66679507 IC50 = 73 nM T47438 C9RS5B 66679618 IC50 = 94 nM T47438 CXN25J 66679626 IC50 = 203 nM T47438 CG5W9J 66679630 IC50 = 1660 nM T47438 C39KZH 66679674 IC50 = 592 nM T47438 CUC7E1 66679703 IC50 = 60 nM T47438 C9VK6Q 66679957 IC50 = 603 nM T47438 C5LTS2 66790999 IC50 = 420 nM T47438 C4DRN2 66791090 IC50 = 660 nM T47438 C0BM4Q 66855521 IC50 = 93 nM T47438 C41HEV 66855843 IC50 = 25 nM T47438 C95TOQ 66855889 IC50 = 447 nM T47438 CGLH60 66856047 IC50 = 270 nM T47438 C74OTM 66856571 IC50 = 5750 nM T47438 C4FE1H 66856796 IC50 = 220 nM T47438 C9LR2W 66856924 IC50 = 6920 nM T47438 C28GNT 66857307 IC50 = 190 nM T47438 CO1IU0 66857459 IC50 = 6170 nM T47438 CE3GP6 66857489 IC50 = 620 nM T47438 CRA3U4 66857678 IC50 = 650 nM T47438 CH79EA 66857904 IC50 = 120 nM T47438 CYPW36 66978859 IC50 = 130 nM T47438 CV4RP5 67281831 IC50 = 69 nM T47438 CXD91K 67282190 IC50 = 363 nM T47438 C7NYX0 67282874 IC50 = 131 nM T47438 C4RH1Q 67282977 IC50 = 133 nM T47438 CMJE32 67282979 IC50 = 18 nM T47438 CK58YL 67283019 IC50 = 2252 nM T47438 C1VB4O 67307922 IC50 > 10000 nM T47438 C48TLF 67308147 IC50 = 930 nM T47438 C52TWL 67308180 IC50 = 70 nM T47438 C5UA6K 67308257 IC50 = 140 nM T47438 CJI01M 67308518 IC50 = 180 nM T47438 C36HRD 67308603 IC50 = 31 nM T47438 CFWV49 67309019 IC50 = 220 nM T47438 C3PV1C 67309038 IC50 = 70 nM T47438 CXEF86 67309051 IC50 = 490 nM T47438 C3UAX0 67309119 IC50 = 1050 nM T47438 C2QA5E 67309143 IC50 = 540 nM T47438 C3RMS8 67309187 IC50 = 120 nM T47438 C8Z3ES 67309205 IC50 = 160 nM T47438 CC4I2B 67309244 IC50 = 170 nM T47438 CU8VA0 67309278 IC50 = 6000 nM T47438 C2NIO8 67309280 IC50 = 660 nM T47438 C7D6AF 67309490 IC50 = 4800 nM T47438 CASD21 67413813 IC50 = 138 nM T47438 CLV4R7 67414480 IC50 = 1216 nM T47438 CP9FJ2 67414954 IC50 = 194 nM T47438 C3G1ZI 67415170 IC50 = 182 nM T47438 CL8FT1 67415210 IC50 = 813 nM T47438 C9K6IY 67415502 IC50 = 339 nM T47438 C4GSO6 67415529 IC50 = 26 nM T47438 CU3E6Y 67415655 IC50 = 78 nM T47438 CF5O8P 67416617 IC50 = 213 nM T47438 CDW41V 67416619 IC50 = 442 nM T47438 CUNK26 67606457 IC50 = 1290 nM T47438 C0MZW4 67606625 IC50 = 500 nM T47438 CL32WA 67606646 IC50 = 8 nM T47438 C9ZJG3 67606672 IC50 = 5 nM T47438 C8CDK5 67606898 IC50 = 135 nM T47438 CV24MS 67606993 IC50 = 710 nM T47438 C49FSK 67607034 IC50 = 52 nM T47438 CQK9F4 67607104 IC50 = 26 nM T47438 CNB15W 67607112 IC50 = 71 nM T47438 CHV08X 67607304 IC50 = 41 nM T47438 C9K5CH 67607317 IC50 = 85 nM T47438 C7N3OX 67607483 IC50 = 280 nM T47438 C37AUI 67607647 IC50 = 27 nM T47438 CT98SM 67607867 IC50 = 11 nM T47438 CX5P7E 67607972 IC50 = 200 nM T47438 C51DEJ 67608037 IC50 = 770 nM T47438 CYX9E6 67608092 IC50 = 45 nM T47438 CVGQ61 67608205 IC50 = 178 nM T47438 CR05TQ 67608430 IC50 = 260 nM T47438 C6FL8Y 67608513 IC50 = 36 nM T47438 CG2OR6 67608703 IC50 = 850 nM T47438 C7Q0LN 67608774 IC50 = 160 nM T47438 CF3S1G 67608840 IC50 = 15 nM T47438 C3PCZ7 67608997 IC50 = 320 nM T47438 CSR21X 67609024 IC50 = 76 nM T47438 C58NAQ 67609354 IC50 = 260 nM T47438 C7H5FX 67609505 IC50 = 603 nM T47438 CPXI26 67700435 IC50 = 1060 nM T47438 CGA89H 68379817 IC50 = 72 nM T47438 CHY40W 68379998 IC50 = 104 nM T47438 C1B6AK 68380073 IC50 = 73 nM T47438 CPA95O 68380152 IC50 = 252 nM T47438 C95VPL 68380260 IC50 = 101 nM T47438 CLBY90 68380304 IC50 = 6 nM T47438 CSC74R 68380314 IC50 = 128 nM T47438 C07ZLW 68380403 IC50 = 302 nM T47438 C02UKY 68380472 IC50 = 15 nM T47438 CM61LR 68495004 IC50 = 580 nM T47438 C0OPQ6 68495695 IC50 = 130 nM T47438 CXU94C 68624921 IC50 = 300 nM T47438 CH5FN4 69491281 IC50 = 140 nM T47438 CC8QU9 70227534 IC50 = 24 nM T47438 CT71PW 70271003 IC50 = 550 nM T47438 CA27SR 70681184 IC50 = 2070 nM T47438 C23CRI 70681196 IC50 = 1090 nM T47438 CH4Z3G 70681292 IC50 = 110 nM T47438 C1UBD3 70683285 IC50 = 300 nM T47438 CJ4P9D 70683379 IC50 = 110 nM T47438 CEZ21F 70683380 IC50 = 90 nM T47438 CNH04A 70685394 IC50 = 7420 nM T47438 CP6KD8 70685475 IC50 = 50 nM T47438 CBO7F4 70685476 IC50 = 210 nM T47438 CR31EK 70685477 IC50 = 120 nM T47438 CK1G2I 70686452 IC50 = 1.04 nM T47438 C3S8PO 70687527 IC50 = 817 nM T47438 CL8W4C 70687532 IC50 = 160 nM T47438 CR73XZ 70687533 IC50 = 420 nM T47438 C85ORZ 70687534 IC50 = 80 nM T47438 CFO9M4 70687535 IC50 = 80 nM T47438 C6JX3Q 70687593 IC50 = 2600 nM T47438 C3JM6F 70687626 IC50 = 190 nM T47438 CTD2H6 70687627 IC50 = 80 nM T47438 CFQ49O 70687628 IC50 = 160 nM T47438 CF6VM9 70687629 IC50 = 80 nM T47438 C6HN4A 70687630 IC50 = 30 nM T47438 C73WJM 70688498 IC50 > 5000 nM T47438 CIE2O6 70689591 IC50 = 330 nM T47438 CHAV16 70689592 IC50 = 70 nM T47438 CMGO80 70689593 IC50 = 290 nM T47438 CP0O2M 70689684 IC50 > 10000 nM T47438 CNMC10 70689685 IC50 = 400 nM T47438 COB0T1 70689686 IC50 = 60 nM T47438 C1FL0M 70689687 IC50 = 50 nM T47438 C2N1MW 70691706 IC50 = 230 nM T47438 C14ZJR 70691707 IC50 = 430 nM T47438 CV1X9D 70691822 IC50 = 70 nM T47438 CR30DQ 70693785 IC50 = 240 nM T47438 C1RM3T 70693787 IC50 = 30 nM T47438 C52LMB 70693791 IC50 = 1330 nM T47438 C6F3YP 70693884 IC50 = 180 nM T47438 CZX6V9 70693885 IC50 = 50 nM T47438 CS35JI 70693886 IC50 = 640 nM T47438 CSQ1U4 70695560 IC50 = 12 nM T47438 CFB1W2 70695912 IC50 = 20 nM T47438 CX1YS3 70695995 IC50 = 120 nM T47438 CLGU94 70695996 IC50 = 970 nM T47438 CNF49O 70696795 IC50 > 5000 nM T47438 CLA17Z 70696796 IC50 > 5000 nM T47438 CMNO49 71192383 IC50 = 8 nM T47438 CU94LC 71260392 EC50 = 90 nM T47438 CD34HG 71450203 IC50 = 6400 nM T47438 C7SX3I 71450567 IC50 = 11500 nM T47438 CYBE17 71452399 IC50 = 17700 nM T47438 C2EI0Q 71452401 IC50 > 160000 nM T47438 CK85SQ 71452402 IC50 = 7300 nM T47438 C01WUF 71453831 IC50 = 16 nM T47438 CWS9B6 71454178 IC50 = 17700 nM T47438 C7E8LW 71455562 IC50 = 46 nM T47438 CZ0FR2 71455918 IC50 > 40000 nM T47438 CN0G2Y 71457197 IC50 = 100 nM T47438 CHA1Y2 71457710 IC50 = 10000 nM T47438 CO3G6C 71457711 IC50 > 40000 nM T47438 CCW60T 71457712 IC50 = 19800 nM T47438 CNI6L3 71457713 IC50 = 4700 nM T47438 C38SKG 71459162 IC50 = 35 nM T47438 CD5H1K 71459215 IC50 = 48 nM T47438 C2Y7EV 71459621 IC50 = 7600 nM T47438 CG1LN5 71459622 IC50 = 11500 nM T47438 C1ER2C 71459623 IC50 > 80000 nM T47438 CE0L8Q 71459624 IC50 = 27600 nM T47438 CUTC89 71461361 IC50 = 27300 nM T47438 CELP71 71461362 IC50 = 38800 nM T47438 CE32BY 71461363 IC50 = 6700 nM T47438 CBO83G 71461364 IC50 = 47600 nM T47438 CZ9YK5 71462725 IC50 = 11 nM T47438 CRQ6N1 71463084 IC50 = 11300 nM T47438 CK46IV 71463085 IC50 = 5400 nM T47438 C6YD9K 71520616 IC50 = 4.5 nM T47438 C2PEI6 71520617 IC50 = 2.7 nM T47438 CJO7I6 71520701 IC50 = 2.1 nM T47438 CE34VC 71520702 IC50 = 1.4 nM T47438 CCF8I9 71520703 IC50 = 4.7 nM T47438 CD9B7C 71520704 IC50 = 4.3 nM T47438 CD64QG 71520705 IC50 = 1.2 nM T47438 C6S3AU 71520806 IC50 = 1.8 nM T47438 CTX49K 71520807 IC50 = 21 nM T47438 C9GUD6 71520808 IC50 = 1.9 nM T47438 C2N5RD 71520810 IC50 = 280 nM T47438 C8TJK7 71520903 IC50 = 25 nM T47438 CN3CI9 71520904 IC50 = 3.5 nM T47438 C45VZB 71524727 IC50 = 10000 nM T47438 C3Z8EL 71524730 IC50 = 10000 nM T47438 C3TYR5 71524781 IC50 = 10000 nM T47438 CLG84N 71540051 IC50 = 43 nM T47438 CL5I0G 71540052 IC50 = 64 nM T47438 CH5N7C 71540152 IC50 = 53 nM T47438 C8NG0Y 71540153 IC50 = 41 nM T47438 C7XN9A 71552168 IC50 = 0.4 nM T47438 C1V5ZC 71552188 IC50 = 39 nM T47438 C6ES2P 71552253 IC50 = 0.4 nM T47438 C3SH2B 71557331 IC50 = 250 nM T47438 CF24JA 71557332 IC50 = 120 nM T47438 CC47DA 71557333 IC50 = 310 nM T47438 C09VTA 71557334 IC50 = 460 nM T47438 C1HS2T 71557500 IC50 = 260 nM T47438 CE9G0B 71557501 IC50 = 29 nM T47438 CS7JM4 71557502 IC50 = 190 nM T47438 C72SHC 71557504 IC50 = 110 nM T47438 C75RON 71557655 IC50 = 200 nM T47438 CURK41 71557656 IC50 = 510 nM T47438 C62QLB 71557817 IC50 = 290 nM T47438 C38SQK 71574724 IC50 > 30000 nM T47438 C0RY5D 71574725 IC50 > 30000 nM T47438 CLPB03 71574822 IC50 > 30000 nM T47438 COV8K9 71574823 IC50 = 2280 nM T47438 CBE97Z 71574913 IC50 > 30000 nM T47438 CK4YB7 71574914 IC50 = 225 nM T47438 C07NVU 71575007 IC50 = 3.16 nM T47438 CPO3K8 71575103 IC50 = 2.47 nM T47438 C27ADL 71623049 EC50 = 67 nM T47438 C1Q9HS 71680619 EC50 = 22 nM T47438 CH0R3N 71680621 EC50 = 46 nM T47438 CI27WN 71716136 IC50 = 78 nM T47438 C1P4JM 71716463 IC50 = 0.402 nM T47438 CD1AG0 71718313 IC50 > 30000 nM T47438 CZT3I5 71718332 IC50 = 10000 nM T47438 CUZ34P 71746393 IC50 = 43 nM T47438 CA6V3F 71746394 IC50 = 2.1 nM T47438 CD4OV3 71746395 IC50 = 0.33 nM T47438 CSU27O 71746396 IC50 = 1.4 nM T47438 C94KHS 71746397 IC50 = 0.18 nM T47438 CQ1UL5 71746584 IC50 = 0.14 nM T47438 CDEN65 72543942 IC50 > 10000 nM T47438 CR9F6I 72543943 IC50 > 10000 nM T47438 C16ZBK 72543944 IC50 = 1450 nM T47438 CC7T5S 72543945 IC50 = 1530 nM T47438 CXC37J 72543946 IC50 = 1350 nM T47438 CO7JZ1 72543947 IC50 > 10000 nM T47438 CSY96R 72544183 IC50 > 10000 nM T47438 CZQ56P 72544184 IC50 > 10000 nM T47438 CW3BR0 72544185 IC50 = 1110 nM T47438 CFA8B5 72544186 IC50 > 10000 nM T47438 CD8Z0S 72544187 IC50 = 2120 nM T47438 C3YST0 72544408 IC50 = 320 nM T47438 C4XR6N 72544409 IC50 > 10000 nM T47438 C6Z9HC 72544410 IC50 = 2130 nM T47438 COQ63R 72544411 IC50 = 820 nM T47438 C3EJ1X 72544412 IC50 > 10000 nM T47438 CV2BY4 72544413 IC50 = 7000 nM T47438 CFLQ91 72544633 IC50 = 570 nM T47438 C3H5VB 72544634 IC50 > 10000 nM T47438 CX7P3D 72544856 IC50 > 10000 nM T47438 CMLI62 72544858 IC50 = 260 nM T47438 C0UPR3 72545078 IC50 > 10000 nM T47438 C3UE9I 72545079 IC50 = 250 nM T47438 C58EVN 72545080 IC50 = 570 nM T47438 C26ABP 72545081 IC50 = 150 nM T47438 C7QIO8 72545318 IC50 = 20 nM T47438 C3PXJ6 72545565 IC50 = 1290 nM T47438 C8JLR9 72545566 IC50 = 150 nM T47438 C34JIF 72545567 IC50 = 650 nM T47438 CA7Y1S 72547022 IC50 > 10000 nM T47438 CW24CT 72547023 IC50 = 2440 nM T47438 C2NCW7 72547024 IC50 > 10000 nM T47438 C7W9JZ 72547025 IC50 > 10000 nM T47438 C1I6VN 72547026 IC50 = 2100 nM T47438 C0Y6IK 72547282 IC50 = 9400 nM T47438 CK50CR 72547283 IC50 = 2750 nM T47438 CZI51W 72547284 IC50 > 10000 nM T47438 C3PTC5 72547285 IC50 > 10000 nM T47438 CY5DQ1 72547286 IC50 = 720 nM T47438 C5XCD4 72547287 IC50 = 280 nM T47438 C4D6PL 72547528 IC50 = 530 nM T47438 CPSB14 72547529 IC50 = 1830 nM T47438 CY91WF 72547530 IC50 = 1260 nM T47438 C48CJQ 72547531 IC50 = 210 nM T47438 CGTC61 72547532 IC50 = 4060 nM T47438 C81YEF 72547533 IC50 > 10000 nM T47438 CE86LF 73345935 IC50 = 1 nM T47438 CWKT40 73345936 IC50 = 60.9 nM T47438 CAF7D6 73345937 IC50 = 133 nM T47438 CA9NC4 73347460 IC50 = 4.6 nM T47438 CPZ91F 73348985 IC50 = 45 nM T47438 CUJ6D8 73350541 IC50 = 117 nM T47438 CG60TJ 73350542 IC50 = 0.3 nM T47438 C30CPA 73350543 IC50 = 47 nM T47438 CP49WL 73352062 IC50 = 0.22 nM T47438 CJ54XQ 73355022 IC50 = 122 nM T47438 CUQ8P7 73355689 IC50 = 62.6 nM T47438 CHAX61 73356579 IC50 = 662 nM T47438 CQ5EP8 73356580 IC50 = 1.86 nM T47438 CYX9E7 73356581 IC50 = 127 nM T47438 CVD9I2 73356582 IC50 = 9.4 nM T47438 C5C7BQ 73441861 EC50 = 14 nM T47438 CFNG54 73441862 EC50 = 9 nM T47438 CE9S7G 73441910 EC50 = 8 nM T47438 C7RAQ4 74538704 IC50 = 2 nM T47438 CC8X5N 75026445 IC50 = 159 nM T47438 CMG4W9 75026446 IC50 = 34 nM T47438 C3S9XM 75593327 EC50 = 50 nM T47438 C0VR9U 76283428 IC50 = 12 nM T47438 CM0CX5 76283429 IC50 = 13 nM T47438 C20YHA 76283431 IC50 = 228 nM T47438 CE2FS3 76283432 IC50 = 5 nM T47438 CHV72I 76283681 IC50 = 25 nM T47438 CT59ZA 76283684 IC50 = 3 nM T47438 CL76SU 76311131 IC50 = 920 nM T47438 C5GQ4Y 76311132 IC50 = 410 nM T47438 CCY61I 76314929 IC50 = 33 nM T47438 CA90TO 76314930 IC50 = 20 nM T47438 CON91Y 76318326 IC50 = 400 nM T47438 C6LD1Z 76318327 IC50 = 1635 nM T47438 C7HW8O 76318328 IC50 = 311 nM T47438 C78SKI 76318329 IC50 = 135 nM T47438 CPN80M 76318550 IC50 = 1.5 nM T47438 CXJT49 76322016 IC50 = 1498 nM T47438 CKX8R9 76325826 IC50 = 12 nM T47438 C1K4DW 76329211 IC50 = 3400 nM T47438 CXTC05 76329212 IC50 = 530 nM T47438 C1T9YD 76329416 IC50 = 23 nM T47438 C63HQJ 76332863 IC50 = 1270 nM T47438 CE47PB 76333057 IC50 = 1 nM T47438 CM1G0K 76336477 IC50 > 15800 nM T47438 CZK4H7 76336685 IC50 = 180 nM T47438 C0H6RM 88313830 IC50 = 790 nM T47438 CNK3Q7 88875492 IC50 = 86 nM T47438 CQ5VJ6 88875808 IC50 = 87 nM T47438 CF67AV 88875879 IC50 = 63 nM T47438 C7ZV5N 89554314 IC50 = 130 nM T47438 CJSP78 89554316 IC50 = 150 nM T47438 C73HFI 89657800 IC50 = 294 nM T47438 C61XRT 89657803 IC50 = 208 nM T47438 C2UX5Q 89657806 EC50 = 347 nM T47438 C5N4FH 89657810 IC50 = 163 nM T47438 CFJ76Q 89657814 EC50 = 1300 nM T47438 CWRS81 89908079 IC50 = 8 nM T47438 C9VQ2W 90174377 IC50 = 112 nM T47438 C14MXT 90667691 IC50 = 100 nM T47438 C4LWC3 90667692 IC50 = 9800 nM T47438 CPMS46 90667839 IC50 = 60 nM T47438 C3O7HA 90667840 IC50 = 600 nM T47438 C2X1ZG 90667841 IC50 = 3100 nM T47438 CAK3F9 90667842 IC50 = 760 nM T47438 C69TWF 90667843 IC50 = 8400 nM T47438 C89UCI 90667844 IC50 = 95 nM T47438 CM0Z9Y 90667845 IC50 = 520 nM T47438 C6WYN1 90667846 IC50 = 260 nM T47438 CER7B8 90667847 IC50 = 1000 nM T47438 CJK62Z 90667848 IC50 = 780 nM T47438 CK7SA3 90667849 IC50 = 1600 nM T47438 CVZ65U 90667850 IC50 = 4600 nM T47438 CYPQ69 90667851 IC50 = 860 nM T47438 CZ7B4N 90667852 IC50 = 590 nM T47438 C8W2RG 90667853 IC50 = 1300 nM T47438 C26GUK 90667854 IC50 = 220 nM T47438 CFXY12 90667855 IC50 = 200 nM T47438 C62PWT 90667856 IC50 = 3000 nM T47438 C8ANE3 90667857 IC50 = 360 nM T47438 C0PGO5 90667858 IC50 = 230 nM T47438 C92COG 90667859 IC50 = 470 nM T47438 C9TW7Y 90667860 IC50 = 47 nM T47438 C7OPI4 90667861 IC50 = 450 nM T47438 CQTM43 90667862 IC50 = 560 nM T47438 CIAD34 90667863 IC50 = 84 nM T47438 CNU18A 90667864 IC50 = 2500 nM T47438 CWEF89 90667865 IC50 = 340 nM T47438 CU7K8Z 90667866 IC50 = 220 nM T47438 CZI63D 91755037 EC50 = 14 nM T47438 CSK6Z1 91844707 IC50 = 14 nM T47438 CK6O3J 92042908 IC50 = 6 nM T47438 CJ23FH 95180362 IC50 = 150 nM T47438 CK02NB 101593793 IC50 = 6250 nM T47438 CGK2W6 118003167 IC50 = 52 nM T47438 CSN6A7 118003183 IC50 = 9 nM T47438 CL0P4E 118003318 IC50 = 389 nM T47438 C2E6WF 118049905 IC50 = 58.5 nM T47438 CDBI46 118049974 EC50 = 105 nM T47438 CW54AG 118049998 IC50 = 30.5 nM T47438 CV3EL4 118050047 IC50 = 25.6 nM T47438 CJ9L0H 118050068 IC50 = 25.4 nM T47438 CA10PR 118050100 IC50 = 72.4 nM T47438 CEQV79 118050174 IC50 = 20.8 nM T47438 CRUP56 118051801 EC50 = 39 nM T47438 C6MQU8 118051925 EC50 = 101 nM T47438 C1SH7T 118054978 IC50 = 54.3 nM T47438 C8L5NJ 118055002 EC50 = 25 nM T47438 C2U9FP 118055004 IC50 = 54.8 nM T47438 CH08WQ 118055008 IC50 = 11.9 nM T47438 CP0CN6 118055017 IC50 = 90 nM T47438 C3PJN1 118055019 IC50 = 56 nM T47438 CT2XV3 118238206 EC50 = 16 nM T47438 CTJN74 118246000 EC50 = 49 nM T47438 CR94TZ 118246257 EC50 = 71 nM T47438 CQH93R 118389830 IC50 = 129 nM T47438 C2E3HO 118389852 IC50 = 13 nM T47438 C50EMF 118389864 IC50 = 4.9 nM T47438 C42MCT 118389887 IC50 = 181 nM T47438 CNC75S 118389896 IC50 = 5.1 nM T47438 C76YWL 118389909 IC50 = 6 nM T47438 CS75HY 118389912 IC50 = 52 nM T47438 CBIR89 118389918 IC50 = 4.9 nM T47438 CN4F6I 118389934 IC50 = 5.6 nM T47438 C24EQN 118389941 IC50 = 801 nM T47438 C70EHC 118389944 IC50 = 53 nM T47438 CT8NU9 118390140 IC50 = 63 nM T47438 CGZP63 118390142 IC50 = 322 nM T47438 C46CPT 118403551 IC50 = 30 nM T47438 CM2NH5 118478848 IC50 = 250.7 nM T47438 CAS3Q9 118717940 IC50 = 25.12 nM T47438 C3GU9R 118717942 IC50 = 1584.89 nM T47438 C6PGA5 118717943 IC50 = 39.81 nM T47438 C7MT5V 118717944 IC50 = 19.95 nM T47438 CX0E4Z 118717945 IC50 = 39.81 nM T47438 CXBW96 118717946 IC50 = 12.59 nM T47438 C5PY4C 118717947 IC50 = 10 nM T47438 CZQB45 118717948 IC50 = 10 nM T47438 C8GVY4 118717949 IC50 = 15848.93 nM T47438 C5N3XM 118717950 IC50 = 19.95 nM T47438 CM1W4V 118717951 IC50 = 316.23 nM T47438 C8ZD5R 118717953 IC50 = 15.85 nM T47438 C2GD7Q 118717957 IC50 = 39.81 nM T47438 CATJ63 118717964 IC50 = 10 nM T47438 CQ42VG 118717965 IC50 = 31.62 nM T47438 C5FS2H 118717970 IC50 = 63.1 nM T47438 C8G0VO 118717971 IC50 = 12.59 nM T47438 C8A2MI 118717972 IC50 = 10000 nM T47438 CAI6Y5 118717973 IC50 = 63.1 nM T47438 CYOM60 118717977 IC50 = 158.49 nM T47438 CT2L5C 118717979 IC50 = 12.59 nM T47438 CZW41X 118717980 IC50 = 19.95 nM T47438 CB3Y8R 118717981 IC50 = 100 nM T47438 C6DLS9 118717982 IC50 = 39.81 nM T47438 C92TQH 118717986 IC50 = 1258.93 nM T47438 CT6MH3 118717989 IC50 = 50.12 nM T47438 CC07RJ 118719411 IC50 = 22 nM T47438 C0S1FZ 118719628 IC50 = 140 nM T47438 C2TWM9 118719629 IC50 = 58 nM T47438 CY0K7Z 118719630 IC50 = 340 nM T47438 CGK38C 118719631 IC50 = 670 nM T47438 CSP43R 118726362 IC50 = 234 nM T47438 CD2E8S 118726363 IC50 = 42 nM T47438 C6WB1O 118726364 IC50 = 19 nM T47438 C87UJQ 118726365 IC50 = 207 nM T47438 CD0CG9 118726366 IC50 = 128 nM T47438 C1O6GD 118726367 IC50 = 96 nM T47438 CX5G2H 118726368 IC50 = 44 nM T47438 CLMU64 118726369 IC50 = 38 nM T47438 CDX1G4 118726370 IC50 = 17 nM T47438 C21WVF 118726371 IC50 = 92 nM T47438 CGC48T 118726372 IC50 = 170 nM T47438 CQB7L8 118726373 IC50 = 361 nM T47438 CFJ1O9 118726374 IC50 = 418 nM T47438 C1KCQ3 118726375 IC50 = 142 nM T47438 CYPG84 118726376 IC50 = 605 nM T47438 CJ6OE8 118726377 IC50 = 22 nM T47438 CLO50Q 118726378 IC50 = 35 nM T47438 CR9NH6 122178430 IC50 = 20 nM T47438 CQ10JD 122178431 IC50 = 85 nM T47438 C80QLF 122186844 IC50 = 5310 nM T47438 CF47TW 122186845 IC50 = 70 nM T47438 CQM3Z7 122186846 IC50 = 110 nM T47438 CKD2V7 122186847 IC50 = 36 nM T47438 C6UGI9 122186848 IC50 = 350 nM T47438 C3MZN1 122186849 IC50 = 310 nM T47438 CE5C9J 122186850 IC50 = 170 nM T47438 C4Y9AM 122186851 IC50 = 62 nM T47438 CE7LZ2 122186852 IC50 = 10000 nM T47438 CS20UJ 122186853 IC50 = 270 nM T47438 C59JBF 122187726 IC50 = 880 nM T47438 CC7W9L 122187727 IC50 = 40 nM T47438 C2N0KO 122187728 IC50 = 240 nM T47438 CRUK02 122187729 IC50 = 70 nM T47438 C7BF8W 122187730 IC50 = 70 nM T47438 C3DX2S 122187798 IC50 = 56 nM T47438 C9VFM5 122187799 IC50 = 11 nM T47438 CR42XN 122187800 IC50 = 210 nM T47438 C4XCP1 122187801 IC50 = 58 nM T47438 CCU2N7 122187802 IC50 = 13 nM T47438 CT2ZJ6 122187803 IC50 = 1490 nM T47438 CGQ8V9 122187804 IC50 = 260 nM T47438 C5W6XS 124351898 EC50 = 40000 nM T47438 CM25EQ 124660563 IC50 = 0.41 nM T47438 CO4Z8M 127025082 IC50 = 1200 nM T47438 CX47HA 127025378 IC50 = 180 nM T47438 CS1CE6 127025655 IC50 = 140 nM T47438 CK2WV4 127028395 IC50 = 35 nM T47438 CN4W1K 127028397 IC50 = 140 nM T47438 CKI9F8 127028409 IC50 = 20 nM T47438 CK79WY 127028410 IC50 = 1800 nM T47438 CD52OH 127028411 IC50 = 50 nM T47438 CP56WJ 127028412 IC50 = 80 nM T47438 C8A4GZ 127028413 IC50 = 120 nM T47438 CZ72JM 127028414 IC50 = 300 nM T47438 C5FZ7T 127028415 IC50 = 1100 nM T47438 CGR4U3 127028416 IC50 = 380 nM T47438 CH4M9N 127028417 IC50 = 1000 nM T47438 C1R8JC 127028418 IC50 = 50 nM T47438 C8W7QS 127028419 IC50 = 190 nM T47438 C1CWF9 127028424 IC50 = 460 nM T47438 CQM96C 127028425 IC50 = 820 nM T47438 CU1CN2 127028426 IC50 = 100 nM T47438 C9R3XB 127028427 IC50 = 200 nM T47438 CZ59BG 127029070 IC50 = 5 nM T47438 C3N8RT 127029071 IC50 = 21 nM T47438 CZBU47 127029072 IC50 = 36 nM T47438 CPY1N6 127029350 IC50 = 56 nM T47438 C3IXT1 127030015 IC50 = 95000 nM T47438 CV10UT 127030331 IC50 = 580 nM T47438 C28VXD 127030332 IC50 = 360 nM T47438 C23GEY 127046417 IC50 = 26000 nM T47438 CY5W9Z 127047958 IC50 > 75000 nM T47438 CCQ7Y5 127053276 IC50 = 135000 nM T47438 CL6O9Z 127053277 IC50 = 85000 nM T47438 C32JOQ 135858933 IC50 = 72 nM T47438 C23LZV 135869398 IC50 = 411 nM T47438 CS56QT 135869399 IC50 = 220 nM T47438 CW6RJ7 135869400 IC50 = 287 nM T47438 CE13WD 135869401 IC50 = 250 nM T47438 C3LP9O 135869402 IC50 = 163 nM T47438 C51QDS 135869403 IC50 = 111 nM T47438 C3ANW7 135869404 IC50 = 88 nM T47438 CU42ZL 135869405 IC50 = 258 nM T47438 C81QEC 135869406 IC50 = 287 nM T47438 C0B6PF 135869407 IC50 = 218 nM T47438 CN4KG1 135869408 IC50 = 301 nM T47438 CW7Q3G 135878222 IC50 = 85 nM T47438 C72FKJ 135878229 IC50 = 92 nM T47438 CB6EV1 135878230 IC50 = 63 nM T47438 CB9M6Z 135878231 IC50 = 158 nM T47438 C19SRN 135878240 IC50 = 91 nM T47438 CTW0K3 135899156 IC50 = 0.65 nM T47438 CBX90O 135910326 IC50 = 3890 nM T47438 C5EC2O 135910327 IC50 = 660 nM T47438 C4AI7G 136030608 IC50 = 4280 nM T47438 C2HP1X 136030609 IC50 = 6740 nM T47438 CCZO92 136030610 IC50 = 3740 nM T47438 CCQ51T 136030757 IC50 = 4870 nM T47438 C0RU6A 136053698 IC50 = 180 nM T47438 C8AZJ9 136069091 IC50 = 20000 nM T47438 C1U8TM 136160538 IC50 = 340 nM T47438 C9QF0C 136199922 IC50 = 171 nM T47438 CDE9Z1 136224008 IC50 = 0.56 nM T47438 CL74HF 136229224 IC50 = 72 nM T47438 C0XLT5 136264485 IC50 = 1 nM T47438 CW83TZ 136626667 IC50 = 36 nM T47438 CPK9S5 136626671 IC50 = 107 nM T47438 C3NG2Q 136626673 IC50 = 25 nM T47438 CZPV15 136626674 IC50 = 117 nM T47438 C2OSQ1 136627167 IC50 = 3981 nM T47438 C0UP1A 137174951 IC50 = 40 nM T47438 CJC95O 138319684 IC50 = 40 nM T47438 CQE13R 138678573 EC50 = 14 nM T47438 CQ5E0B 138678593 EC50 = 111 nM T47438 C8QH0O 138678605 EC50 = 34 nM T47438 C7H9KZ 138678606 EC50 = 19 nM T47438 C1FZ7S 138678620 EC50 = 35 nM T47438 CLHK06 138678794 EC50 = 36 nM T47438 C2AOQ9 139415485 EC50 = 5 nM T47438 CCT8G2 139415505 EC50 = 8 nM T47438 C3K2ZI 139415517 EC50 = 13 nM T47438 C75SJT 139415533 EC50 = 15 nM T47438 CH62KO 139415536 EC50 = 8 nM T47438 CDM5L3 139415543 EC50 = 33 nM T47438 C0M5IB 139415544 EC50 = 7 nM T47438 C6VF5T 139430688 EC50 = 30 nM T47438 CT1L7K 142606858 IC50 = 14 nM T47438 C0RAK9 142606862 IC50 = 8 nM T47438 CQL72N 142606863 IC50 = 25 nM T47438 CZ4W2M 142606877 IC50 = 49 nM T47438 C65IWN 142606880 IC50 = 27 nM T47438 CG23NY 142606884 IC50 = 16 nM T47438 C1GD8S 142606886 IC50 = 44 nM T47438 CZW98E 142606887 IC50 = 15 nM T47438 C4YPQ7 142606891 IC50 = 23 nM T47438 CO70HU 142606893 IC50 = 31 nM T47438 CU6SN1 142606894 IC50 = 15 nM T47438 C94CBQ 142606895 IC50 = 14 nM T47438 CXV31J 142606896 IC50 = 26 nM T47438 C05MIP 142607769 IC50 = 120 nM T47438 C1LR5J 142607770 IC50 = 1200 nM T47438 C3TMR0 142607778 IC50 = 90 nM T47438 CMFQ84 142607794 IC50 = 2770 nM T47438 C0VR9Y 142607800 IC50 = 350 nM T47438 CE1B9H 142607803 IC50 = 3400 nM T47438 C34GVD 142607804 IC50 = 200 nM T47438 CZYG08 142607806 IC50 = 30 nM T47438 C7MUQ2 142607808 IC50 > 30000 nM T47438 C8TM1A 142607812 IC50 = 70 nM T47438 CO08KN 142607816 IC50 = 40 nM T47438 CPHZ53 142607820 IC50 = 194 nM T47438 CR01WI 142607828 IC50 > 30000 nM T47438 CDZ91R 142607841 IC50 = 60 nM T47438 CN09SF 142607846 IC50 = 730 nM T47438 CL3D6V 142607847 IC50 = 1390 nM T47438 CF79IB 142607849 IC50 = 4570 nM T47438 CA8TY4 142607851 IC50 = 200 nM T47438 C5A1MS 142607854 IC50 = 3130 nM T47438 CY6FI1 142607870 IC50 = 680 nM T47438 CBX8T3 142607871 IC50 = 750 nM T47438 C3B0JS 142607879 IC50 = 670 nM T47438 CBD2L5 142607880 IC50 = 430 nM T47438 CU39BH 142607882 IC50 = 50 nM T47438 C7KTU5 142607897 IC50 = 740 nM T47438 C73HXD 142607900 IC50 = 380 nM T47438 CZ91AK 145955876 IC50 = 21700 nM T47438 CS6Z9D 145961223 IC50 = 180 nM T47438 CHR50A 145961243 IC50 = 60 nM T47438 CQ0YK2 145961280 IC50 = 500 nM T47438 C6ID3H 145961522 IC50 = 2200 nM T47438 CSB5U8 145961774 IC50 = 60 nM T47438 CWI9B1 145961933 IC50 = 20 nM T47438 CWB80D 145962590 IC50 = 40 nM T47438 CJ5A6Q 145962645 IC50 = 950 nM T47438 C4H9TL 145963152 IC50 = 160 nM T47438 CE7UM2 145963197 IC50 = 70 nM T47438 CCRH49 145963599 IC50 = 9 nM T47438 CIQ30C 145963822 IC50 > 50000 nM T47438 C5E3FO 145964932 IC50 = 690 nM T47438 CC9QL4 145966531 IC50 = 1800 nM T47438 CQV46Y 145970305 IC50 = 17 nM T47438 CDTU34 145970496 IC50 > 10000 nM T47438 CKH7U4 145972721 IC50 = 1300 nM T47438 CJ0US7 145973873 IC50 = 7100 nM T47438 C2SQV7 145974463 IC50 = 390 nM T47438 C0DWZ2 145976055 IC50 = 9800 nM T47438 CVF1G3 145977207 IC50 = 5800 nM T47438 CFZA28 145977593 IC50 > 50000 nM T47438 CEX8V9 145978454 IC50 = 8700 nM T47438 C4HQO0 145978536 IC50 = 2300 nM T47438 CO5RK9 145988561 EC50 = 14 nM T47438 CLO3W7 145992890 EC50 = 8 nM T47438 C73LTZ 146306592 EC50 = 0.013 nM T47438 CD6KR9 146306602 EC50 = 0.0103 nM T47438 C7O4XE 146306604 EC50 = 0.0114 nM T47438 CR9V2L 146306617 EC50 = 0.0117 nM T47438 CT3H9B 146306631 EC50 = 0.0059 nM T47438 CO69MS 155164669 IC50 = 39 nM T47438 CQ1EW0 155510983 EC50 = 10 nM T47438 CT4LJ1 155512934 IC50 = 41 nM T47438 C24AKY 155513525 IC50 = 175 nM T47438 C2DSZ8 155513622 EC50 = 6 nM T47438 COQX09 155515761 IC50 > 1000 nM T47438 C94IPH 155517286 IC50 = 110 nM T47438 CVAI54 155517459 EC50 = 20 nM T47438 CKZ7Y8 155518783 IC50 = 45 nM T47438 C5QGD4 155519995 IC50 = 98 nM T47438 C1AZB0 155520838 IC50 = 475 nM T47438 CIC5L7 155521256 IC50 = 603 nM T47438 C3KSY8 155522962 EC50 = 45 nM T47438 CRH81M 155523684 IC50 = 179 nM T47438 CFA5X1 155524819 IC50 = 362 nM T47438 CQXZ91 155525880 IC50 = 114 nM T47438 CAM48S 155526231 EC50 = 0.0092 nM T47438 C69CBF 155526641 IC50 = 18 nM T47438 CD5QT6 155526690 IC50 > 1000 nM T47438 C50HCX 155526887 IC50 = 216 nM T47438 CC1O5K 155530531 IC50 = 49 nM T47438 CUW4Z9 155530939 IC50 = 394 nM T47438 CSU48Z 155531407 IC50 = 148 nM T47438 CFL61W 155532250 IC50 = 19 nM T47438 CE8Y0F 155532723 IC50 = 112 nM T47438 C18XWC 155533276 IC50 = 225 nM T47438 C0PD6N 155533341 IC50 = 219 nM T47438 CM6HK5 155533472 IC50 = 55 nM T47438 C2QHX4 155534806 IC50 = 15 nM T47438 CB63DW 155539872 IC50 = 771 nM T47438 CXIS50 155540564 IC50 = 280 nM T47438 C8AJU4 155540955 IC50 > 1000 nM T47438 C4RUM6 155542247 IC50 = 31 nM T47438 C6IVD9 155542803 IC50 = 23 nM T47438 C0TDZ4 155544576 IC50 = 270 nM T47438 CEY5H1 155544970 IC50 = 87 nM T47438 C0F3HL 155546703 IC50 = 4000 nM T47438 CG50LE 155547624 IC50 > 1000 nM T47438 CA5ID2 155547685 IC50 = 110 nM T47438 CV9LR8 155547786 IC50 = 39 nM T47438 C65HFR 155547882 EC50 = 0.0139 nM T47438 CB9V6O 155548351 EC50 = 21 nM T47438 C27AGI 155549080 EC50 = 6 nM T47438 C9H8MJ 155549445 IC50 = 26 nM T47438 CXQR20 155550079 IC50 = 195 nM T47438 CS5GJ8 155550249 IC50 = 67 nM T47438 C02QZK 155551379 IC50 = 62 nM T47438 CTP2Z9 155551650 IC50 = 36 nM T47438 CNBK91 155552409 IC50 = 32 nM T47438 C9IOT0 155553367 IC50 > 1000 nM T47438 C1GI7C 155554967 IC50 = 66 nM T47438 C4SGF5 155556571 EC50 = 41 nM T47438 C3HMY5 155557465 IC50 = 66 nM T47438 C1SVN7 155558409 IC50 = 41 nM T47438 C0TK7L 155558815 IC50 = 289 nM T47438 CVP1I3 155559282 IC50 = 85 nM T47438 C56CPG 155559540 IC50 = 17 nM T47438 CY05DH 155560260 IC50 = 92 nM T47438 CI5JV9 155560962 IC50 = 94 nM T47438 CV3RC0 155561296 IC50 > 1000 nM T47438 C8NA0K 155562228 IC50 = 347 nM T47438 CR7TI5 155562738 IC50 = 229 nM T47438 C1XZM9 155563081 IC50 = 110 nM T47438 C2H5JE 155565668 IC50 > 1000 nM T47438 CH39OK 155565786 IC50 = 766 nM T47438 CT4GP1 155566638 IC50 = 22 nM T47438 C0CRB1 155567585 IC50 = 121 nM T47438 CM4XS2 155567732 EC50 = 0.0064 nM T47438 C2BDR8 155568466 IC50 = 59 nM T47438 CGWF78 155568726 IC50 = 272 nM T47438 CKYJ21 76283430 IC50 = 6 nM T47438 CIJ3N0 76283682 IC50 = 23.3 nM T47438 D00DFR 11809004 IC50 = 1100 nM T47438 D03AMR 9849669 IC50 = 200 nM T47438 D04TWU 15071517 IC50 = 6900 nM T47438 D0B5FC 447912 EC50 = 3600 nM T47438 D0I8BA 16037828 IC50 = 1000 nM T47438 D0K8LN 44400752 IC50 = 461 nM T47438 D0M2LV 44413811 IC50 = 4900 nM T47438 D0Q6ZQ 53308121 IC50 = 5.3 nM T02226 D00MXN 25019940 Ki = 0.021 nM T02226 D0G5ME 11319053 Ki = 0.77 nM T02226 D0IA9Y 53472683 Ki = 0.023 nM T02226 D0L5GH 6918509 Ki = 0.01 nM T02226 D0V9VG 51049968 Ki = 0.027 nM T02226 CW2XB1 9978597 Ki = 78 nM T02226 CSY53V 10077700 Ki = 0.012 nM T02226 C9RXY3 10102983 IC50 = 146 nM T02226 CEP07A 10340395 Ki = 280 nM T02226 CC36IR 10340456 Ki = 309 nM T02226 C0EQX7 10394458 Ki = 0.011 nM T02226 C01PKW 10416497 IC50 = 0.074 nM T02226 C0YSQ7 10416713 Ki = 0.005 nM T02226 C4S2JZ 10433192 IC50 = 5500 nM T02226 C69MPT 10438558 IC50 = 3.2 nM T02226 CS94QC 10453991 Ki = 607 nM T02226 CXP35B 10483468 IC50 = 87 nM T02226 CHNT90 10483685 Ki = 32 nM T02226 CFG4O3 11156698 IC50 = 4.4 nM T02226 CSQP28 11157609 Ki = 6900 nM T02226 CFC0L9 11157626 IC50 = 224 nM T02226 C1R4CH 11158071 Ki = 0.22 nM T02226 C0KY1X 11168000 Ki = 11 nM T02226 C8BLU1 11169408 IC50 = 1.9 nM T02226 C6Q9MF 11169454 IC50 = 0.34 nM T02226 C1TY6Q 11180666 Ki = 1.7 nM T02226 CR4O1G 11191890 IC50 = 10 nM T02226 CXF10W 11192602 Ki = 0.5 nM T02226 CV6NF8 11192748 IC50 = 1.3 nM T02226 CKE6B8 11204498 IC50 = 0.19 nM T02226 CTS40R 11204595 Ki = 0.039 nM T02226 CQI1R0 11215322 Ki = 427 nM T02226 CNL48A 11215412 IC50 = 12 nM T02226 CJ39MV 11215446 IC50 = 0.49 nM T02226 CA7H8W 11215502 Ki = 983 nM T02226 CNW94U 11215639 Ki = 6400 nM T02226 C6BZ8W 11225752 Ki = 2.7 nM T02226 C2U7FL 11226747 IC50 = 1.4 nM T02226 CAY0X1 11227287 Ki > 10000 nM T02226 C2I7CU 11238250 IC50 = 28 nM T02226 CJD59I 11238677 IC50 = 0.42 nM T02226 C7GZ9Q 11238717 Ki = 2800 nM T02226 CSZ2M3 11249157 IC50 = 30 nM T02226 C7J4WT 11250445 IC50 = 0.63 nM T02226 CMX8H7 11250446 IC50 = 0.98 nM T02226 CT2KR7 11261842 Ki = 965 nM T02226 C39NJZ 11273798 IC50 = 4.8 nM T02226 C1I4RB 11284233 Ki = 0.9 nM T02226 CL41QP 11286085 IC50 = 776.25 nM T02226 CF65RC 11295168 IC50 = 3.1 nM T02226 CGPS72 11295951 IC50 = 0.46 nM T02226 C3HZ9A 11297807 IC50 = 588.84 nM T02226 CHM45S 11308069 IC50 = 0.099 nM T02226 CKQ01L 11308219 IC50 = 0.089 nM T02226 CXF31N 11330650 Ki = 685 nM T02226 CGML40 11330786 Ki = 320 nM T02226 C6TFR2 11341430 IC50 = 3.8 nM T02226 CAV4B2 11341642 IC50 = 0.94 nM T02226 CR9J6K 11342207 Ki = 853 nM T02226 CKTZ78 11351794 Ki = 22 nM T02226 C2SN5F 11354531 Ki = 0.14 nM T02226 C7L3VT 11364682 IC50 = 0.21 nM T02226 CPV21T 11364735 Ki = 0.3 nM T02226 C89EDQ 11365194 IC50 = 1583 nM T02226 CR6H4L 11375693 Ki = 2.4 nM T02226 CM87TN 11375696 IC50 = 120 nM T02226 C18WDP 11377534 Ki = 0.023 nM T02226 CR2F7Y 11387141 IC50 = 2.1 nM T02226 CJ7U4X 11387595 Ki = 0.9 nM T02226 CGY80S 11388586 Ki = 0.055 nM T02226 C4YTL3 11397560 Ki = 3.6 nM T02226 CJ7B1C 11398863 IC50 = 4.8 nM T02226 CZQ35I 11409395 IC50 = 97 nM T02226 CB6TC2 11410749 IC50 = 34 nM T02226 CJ1CM9 11411030 IC50 = 0.39 nM T02226 CTV17E 11421827 Ki = 22 nM T02226 C54GDM 11422298 IC50 = 0.078 nM T02226 CZU3S7 11423175 IC50 = 4466.84 nM T02226 C0YT2F 11432183 IC50 = 8.6 nM T02226 CHGT51 11432505 Ki = 10 nM T02226 C6CE9W 11432931 Ki = 0.7 nM T02226 CYZ92S 11434781 IC50 = 707.95 nM T02226 C3B2TE 11443894 IC50 = 35 nM T02226 C56IND 11444574 IC50 = 7.4 nM T02226 CRE9W2 11444589 Ki = 156 nM T02226 CAI0X1 11444699 Ki = 6100 nM T02226 C62PUD 11445240 Ki = 0.28 nM T02226 C6CD1Y 11453687 Ki = 83 nM T02226 C2MOP7 11454113 Ki = 51 nM T02226 CW5BO3 11456078 IC50 = 1.6 nM T02226 CJU06L 11456102 Ki = 295 nM T02226 CH6S7Z 11456201 IC50 = 0.88 nM T02226 C1U8CX 11466363 IC50 = 1.5 nM T02226 CY1EG6 11467108 IC50 = 1 nM T02226 C16NBP 11467753 Ki = 0.0073 nM T02226 CFOC05 11478841 IC50 = 0.83 nM T02226 CFC93K 11478962 IC50 = 0.13 nM T02226 CHF3T7 11495985 IC50 = 495 nM T02226 C9WD3C 11497403 Ki = 855 nM T02226 C0P1QE 11498219 IC50 = 0.02 nM T02226 CN2Y7Z 11505361 Ki = 2000 nM T02226 C01MDL 11512851 IC50 = 0.063 nM T02226 CQUV12 11512928 Ki = 1.1 nM T02226 CV92TG 11513230 IC50 > 300000 nM T02226 C4D0FS 11519899 Ki = 110 nM T02226 CT97KM 11520007 Ki = 0.63 nM T02226 CFDQ43 11520022 Ki = 339 nM T02226 C8EI9U 11520204 IC50 = 0.057 nM T02226 CDG8W2 11526993 Ki = 3.5 nM T02226 C5TFH3 11527287 Ki = 720 nM T02226 CU8CE9 11532845 Ki = 96 nM T02226 CHF2N8 11534977 IC50 = 17000 nM T02226 CAD16K 11541560 Ki = 1.1 nM T02226 CJ6E4C 11541725 Ki = 27 nM T02226 CHS87Q 11548734 IC50 = 23 nM T02226 C7SK0A 11549001 IC50 = 450 nM T02226 C9HT8K 11549159 IC50 = 0.022 nM T02226 CR79TM 11555955 Ki = 46 nM T02226 CEK1F3 11562434 Ki = 3.7 nM T02226 C8DIQ5 11570464 Ki = 5337 nM T02226 C20RJY 11570753 Ki = 1050 nM T02226 CE4IT9 11571094 Ki = 19 nM T02226 CP8M4A 11576078 Ki = 270 nM T02226 CA9TQ4 11578671 IC50 = 17000 nM T02226 C18FPK 11584808 Ki = 1.7 nM T02226 C9LQD0 11585317 Ki = 6.3 nM T02226 CG4FL3 11592648 IC50 = 0.068 nM T02226 CCAQ30 11599135 IC50 = 1.8 nM T02226 C4O7JT 11599531 IC50 = 120 nM T02226 C4X7NH 11599798 IC50 = 0.053 nM T02226 C30LBG 11599872 IC50 = 0.13 nM T02226 CO0V9M 11599913 IC50 = 0.011 nM T02226 CNU10O 11606400 Ki = 0.69 nM T02226 CBV9D3 11621504 IC50 = 0.01 nM T02226 CNT8V6 11628731 Ki = 11 nM T02226 C7Z4AE 11636224 IC50 > 300000 nM T02226 CWE5X4 11650307 IC50 = 193 nM T02226 CK3UO8 11657395 IC50 = 0.044 nM T02226 C08UGA 11671386 Ki = 2900 nM T02226 C9B6GR 11678239 Ki = 3.2 nM T02226 CO4DL5 11678456 Ki = 20000 nM T02226 C1JFI5 11685954 IC50 = 0.017 nM T02226 CX4Q2U 11691938 Ki = 3.1 nM T02226 C69HMB 11692140 Ki = 4 nM T02226 C87ZSQ 11692206 Ki = 583 nM T02226 CO3EI9 11692628 Ki = 1.1 nM T02226 C4XFK0 11693761 IC50 = 44 nM T02226 C29VOY 11699891 Ki = 3.9 nM T02226 CVLK50 11706251 Ki = 46 nM T02226 CG0B5Q 11706981 Ki = 0.07 nM T02226 C8RCQ9 11707040 Ki = 11 nM T02226 C7XJ8D 11713729 Ki = 575 nM T02226 C2NC5F 11713849 Ki = 1249 nM T02226 CF76KX 11721278 Ki = 1.1 nM T02226 CW8V7S 11752904 Ki = 1.4 nM T02226 C24ODM 11753021 Ki = 1.4 nM T02226 CX19UV 11753024 IC50 = 6 nM T02226 C1EMS2 11785573 IC50 = 4.8 nM T02226 CB17JY 11785754 IC50 = 12 nM T02226 C01QPC 11786529 Ki = 51 nM T02226 CE0HF8 11786642 IC50 = 0.38 nM T02226 C5RPV6 11848645 Ki = 220 nM T02226 CY6X8K 11848646 Ki = 43 nM T02226 C81SEQ 11848647 Ki = 270 nM T02226 C1PN7A 11848698 Ki = 9000 nM T02226 C0NF3B 11848750 Ki = 75 nM T02226 CHL78I 11848753 Ki = 1750 nM T02226 CL4S1Z 11848755 Ki = 495 nM T02226 C7KZL1 11848798 Ki = 1900 nM T02226 C9EAL0 11848800 Ki = 228 nM T02226 CPSU54 11848855 Ki = 74 nM T02226 CNP83T 11848857 Ki = 695 nM T02226 CWRO47 11848908 Ki = 41 nM T02226 C23ZVT 11848963 Ki = 170 nM T02226 C67WMH 11848964 Ki = 95 nM T02226 C8K9IP 11848965 Ki = 54 nM T02226 C9E7VN 11848966 Ki = 42 nM T02226 CHM18G 11848968 Ki = 105 nM T02226 C4ZY7K 11849020 Ki = 96 nM T02226 C4VI7D 11849023 Ki = 635 nM T02226 CS17WY 11849024 Ki = 205 nM T02226 C1LYJ0 11849025 Ki = 17 nM T02226 C21UVM 11849147 Ki = 80 nM T02226 CUT84W 16115156 IC50 = 107.15 nM T02226 C2I4RM 16745090 Ki = 185 nM T02226 CR79HP 21102037 IC50 = 2 nM T02226 CK10IC 21102038 IC50 = 3.7 nM T02226 CZ1Q0N 21102224 EC50 = 31 nM T02226 C9FW6Z 23627980 Ki = 35 nM T02226 CLQ2B0 23654987 Ki = 0.3 nM T02226 CAH83C 23656586 Ki = 4400 nM T02226 CE4ZM7 23656587 Ki = 770 nM T02226 CYKB10 23656588 Ki = 9900 nM T02226 CWMD21 23656749 Ki = 470 nM T02226 CBS03U 23656750 Ki = 1700 nM T02226 CRET24 23656751 Ki = 1100 nM T02226 CGR12U 23656752 Ki = 470 nM T02226 CCE3B5 23656753 Ki = 610 nM T02226 C7CO2B 23656918 Ki = 37 nM T02226 C3JIP1 23656919 Ki = 93 nM T02226 CDL81I 23656920 Ki = 4.2 nM T02226 CRQ31C 23656921 Ki = 0.19 nM T02226 CV96FP 23656922 Ki = 4.9 nM T02226 CM27YU 23657089 Ki = 0.5 nM T02226 CH2L9G 24756611 EC50 = 12 nM T02226 CVG14A 24756612 EC50 = 130 nM T02226 C7DL3K 24756690 IC50 = 0.33 nM T02226 CF3J6T 24756767 IC50 = 5.9 nM T02226 CF40KL 24756768 IC50 = 34 nM T02226 CQ3X4L 24756769 IC50 = 15 nM T02226 C3X4NK 24756770 IC50 = 460 nM T02226 C08WIS 24853163 Ki = 88 nM T02226 CZK38U 24853164 Ki = 2 nM T02226 CJ4T7O 24853374 Ki = 32 nM T02226 CO73CZ 24862842 Ki = 68 nM T02226 C0UN7H 24863246 Ki = 28 nM T02226 C84JXU 24863323 Ki = 0.55 nM T02226 CUY1O2 24863332 Ki = 0.27 nM T02226 CV29XP 24863333 Ki = 0.23 nM T02226 CJIN21 24863334 Ki = 0.65 nM T02226 CAFZ85 25019993 Ki = 0.034 nM T02226 C0X8DC 25034109 Ki = 0.55 nM T02226 CY8EP0 25110584 Ki = 6.31 nM T02226 CURE82 25151777 Ki = 3.981 nM T02226 CSP1W0 25151968 Ki = 3.162 nM T02226 CUM6S8 25152167 Ki = 5.012 nM T02226 C78MVE 25152169 Ki = 2.512 nM T02226 CYR8F9 25152367 Ki = 7.943 nM T02226 CP0U4K 25152370 Ki = 12.59 nM T02226 CWI75J 25152560 Ki = 15.85 nM T02226 CN8BM0 25152561 Ki = 25.12 nM T02226 C2OB9H 25152563 Ki = 125.89 nM T02226 CP0W7T 25152564 Ki = 125.89 nM T02226 C3ZWB2 25152765 Ki = 6.31 nM T02226 C0EL1C 25152766 Ki = 3.981 nM T02226 C2K3LX 25152981 Ki = 50.12 nM T02226 C3BI5L 25152984 Ki = 25.12 nM T02226 CA64HU 25152985 Ki = 25.12 nM T02226 C8LK9M 25153832 Ki = 1.585 nM T02226 C9TA6K 25154032 Ki = 3.981 nM T02226 C9MW8O 25154034 Ki = 2.512 nM T02226 C2KTS7 25181509 Ki = 0.039 nM T02226 CIM67A 25227362 Ki = 0.51 nM T02226 CHRS21 44273362 IC50 = 70000 nM T02226 CM4PQ5 44273364 IC50 = 51000 nM T02226 CVSZ14 44273516 IC50 > 100000 nM T02226 CDX27H 44273596 IC50 = 8550 nM T02226 CS53AM 44273608 IC50 = 5000 nM T02226 C3S5NZ 44273609 IC50 = 95000 nM T02226 C24FZC 44273610 IC50 = 7000 nM T02226 CP48DY 44273621 IC50 = 6900 nM T02226 C83HLE 44273622 IC50 = 4275 nM T02226 CDU4K9 44273716 IC50 > 3000 nM T02226 CTO2F1 44273717 IC50 > 3000 nM T02226 C93UJI 44273718 IC50 = 220 nM T02226 CIP61B 44273804 IC50 = 3000 nM T02226 CC02NK 44273825 IC50 = 10000 nM T02226 CCG57H 44273826 IC50 = 10000 nM T02226 C2K8FX 44273827 IC50 = 10000 nM T02226 C3BYF4 44273842 IC50 = 45000 nM T02226 C20HDP 44273843 IC50 > 100000 nM T02226 CIX61G 44273844 IC50 = 200 nM T02226 CIE3V4 44273845 IC50 > 10000 nM T02226 CHB1T0 44273857 IC50 = 360 nM T02226 C1E0JP 44273858 IC50 = 470 nM T02226 C12THF 44273867 IC50 = 9000 nM T02226 CVE0I8 44273868 IC50 = 300 nM T02226 CS2EI3 44273869 IC50 = 8000 nM T02226 C6DU4X 44273870 IC50 = 24000 nM T02226 CIU4V7 44273871 IC50 = 10000 nM T02226 C1AP7W 44273878 IC50 = 1200 nM T02226 C9Z1IG 44273880 IC50 = 2700 nM T02226 CJG5M9 44273881 IC50 = 6500 nM T02226 CB8NE4 44273909 IC50 = 4000 nM T02226 C4BUD5 44273948 IC50 > 10000 nM T02226 CNRA07 44273949 IC50 = 3400 nM T02226 CBCP21 44273950 IC50 = 32000 nM T02226 C7X1FO 44273967 IC50 = 24000 nM T02226 CAO4P7 44273969 IC50 > 100000 nM T02226 CD7J9B 44273976 IC50 = 490 nM T02226 C0ZBP1 44273979 IC50 = 280 nM T02226 CA02ZL 44273980 IC50 > 10000 nM T02226 CR54UE 44273987 IC50 = 18000 nM T02226 CVM9S8 44273992 IC50 = 80000 nM T02226 CQE3U0 44273994 IC50 = 4790 nM T02226 C36GES 44274008 IC50 = 10000 nM T02226 C6JCG2 44274013 IC50 > 10000 nM T02226 CG0A2V 44274014 IC50 = 4500 nM T02226 CXCT49 44274025 IC50 = 620 nM T02226 C02GLR 44274032 IC50 = 205 nM T02226 CO60FW 44274035 IC50 = 10000 nM T02226 C93URN 44274036 IC50 = 10000 nM T02226 CQ5O3Z 44274037 IC50 = 14000 nM T02226 CV3A8Z 44274039 IC50 > 10000 nM T02226 C0WQV6 44274073 IC50 = 10000 nM T02226 CGJ56K 44274074 IC50 > 100000 nM T02226 C6Z9AJ 44274076 IC50 > 100000 nM T02226 C5Y7LE 44274096 IC50 > 3000 nM T02226 CV17HE 44274097 IC50 > 10000 nM T02226 CNO3Y6 44274098 IC50 = 170 nM T02226 C98IRQ 44274099 IC50 = 4500 nM T02226 CXVF03 44274101 IC50 = 3000 nM T02226 CBYZ92 44323001 IC50 = 17000 nM T02226 CG2WX7 44323086 IC50 > 100000 nM T02226 C0KZ2L 44323087 IC50 > 100000 nM T02226 C0Q6DS 44323095 IC50 = 5200 nM T02226 C6G1KZ 44323097 IC50 = 12000 nM T02226 C64YGA 44323110 IC50 = 96000 nM T02226 CD2S7Q 44323139 IC50 = 33000 nM T02226 CIO08E 44323180 IC50 = 9900 nM T02226 CC4YF1 44323332 IC50 = 41000 nM T02226 CFAY53 44323338 IC50 = 37000 nM T02226 C12WJT 44323339 IC50 > 100000 nM T02226 C5OGN1 44323341 IC50 = 74000 nM T02226 C49QHD 44403853 IC50 = 13000 nM T02226 C4TF8U 44403854 IC50 = 1000 nM T02226 C3AU1P 44403855 IC50 = 200 nM T02226 CZJ63F 44403856 IC50 = 226 nM T02226 CWS0U9 44403857 IC50 = 250 nM T02226 C1LW2J 44403858 IC50 = 44 nM T02226 C3X7GN 44403859 IC50 = 4.7 nM T02226 CJK6A8 44403860 IC50 = 0.2 nM T02226 CU3C1O 44403861 IC50 = 0.03 nM T02226 CNR30J 44403862 IC50 = 0.05 nM T02226 CJ6PA5 44403914 IC50 = 50000 nM T02226 C15ZXC 44403915 IC50 > 300000 nM T02226 CF24BX 44403916 IC50 > 300000 nM T02226 CUDT41 44403917 IC50 = 10300 nM T02226 CSA8I5 44403918 IC50 = 196000 nM T02226 CIR8W1 44404069 IC50 = 40000 nM T02226 CJ69ZX 44416436 IC50 = 373 nM T02226 C9X3NK 44416437 Ki = 143 nM T02226 CWYX41 44416442 Ki = 1000 nM T02226 C0GQL1 44416488 Ki = 3800 nM T02226 C2UHG0 44416512 IC50 = 715 nM T02226 C7JI1G 44416513 Ki = 1055 nM T02226 C1ZM4Q 44416514 IC50 = 220 nM T02226 C5HIN3 44416516 Ki = 20000 nM T02226 CXY19R 44416912 Ki = 11 nM T02226 CDS7E4 44417049 Ki = 104 nM T02226 CODP98 44417050 Ki = 27 nM T02226 CQO2U8 44420227 Ki = 87 nM T02226 CAM5F1 44420228 Ki = 38 nM T02226 C5LB7G 44420231 Ki = 29 nM T02226 CY2F3Q 44420235 Ki = 20 nM T02226 C46VUS 44420236 Ki = 8.7 nM T02226 CC9MN0 44420240 Ki = 20 nM T02226 CM89QF 44420241 Ki = 6.8 nM T02226 C4V5SX 44420245 Ki = 15 nM T02226 CO9BH3 44420250 Ki = 10 nM T02226 C7ANU1 44420255 Ki = 25 nM T02226 C8TE2M 44420256 Ki = 12 nM T02226 CL2FN9 44420260 Ki = 9.5 nM T02226 CFWC52 44420261 Ki = 17 nM T02226 C1T6IE 44420286 Ki = 103 nM T02226 CFPY38 44420287 Ki = 48 nM T02226 C3NQT1 44420290 Ki = 1050 nM T02226 CZY17T 44420691 IC50 = 380.19 nM T02226 C3H1EF 44420692 IC50 = 67.61 nM T02226 CWX81Y 44420693 IC50 = 5754.4 nM T02226 CZS90I 44421021 EC50 = 0.2 nM T02226 C0NAY5 44454954 Ki = 390 nM T02226 CLV3J4 44455041 Ki = 166 nM T02226 CPS61E 44455043 Ki = 155 nM T02226 CY4N5D 44455078 Ki = 213 nM T02226 CY7OU8 44455080 Ki = 71 nM T02226 CECP81 44455153 Ki = 42 nM T02226 CJQ05D 44455188 Ki = 2050 nM T02226 CJ81LT 44455348 Ki = 3400 nM T02226 CXUZ08 44455457 Ki = 140 nM T02226 CB5T0Z 44468576 Ki = 0.094 nM T02226 C9C1RH 44468711 Ki = 0.5 nM T02226 CS2AV5 44469523 Ki = 0.11 nM T02226 C91APQ 44469664 Ki = 0.019 nM T02226 C31OVU 44469946 Ki = 0.021 nM T02226 C63BGP 44470090 Ki = 0.045 nM T02226 CVR8Q5 44562895 Ki = 5.5 nM T02226 CMRN61 44562896 Ki = 41 nM T02226 CYR7O0 44562897 Ki = 13 nM T02226 C9J2TE 44562936 Ki = 32 nM T02226 CG6A2F 44562937 Ki = 26 nM T02226 C2JZI8 44562938 Ki = 100 nM T02226 C35UFM 44562939 Ki = 15 nM T02226 CMI43S 44562982 Ki = 18 nM T02226 CZ2IV8 44562983 Ki = 62 nM T02226 C7XS9M 44562984 Ki = 23 nM T02226 CKA21W 44562985 Ki = 9.5 nM T02226 CQ8NJ3 44563025 Ki = 15 nM T02226 CPE7L6 44563026 Ki = 120 nM T02226 C8BMF5 44563027 Ki = 250 nM T02226 CV8BX9 44563028 Ki = 2.7 nM T02226 CFS8T3 44563050 Ki = 2.1 nM T02226 C5GLD7 44563051 Ki = 21 nM T02226 C0MX4G 44563052 Ki = 1.9 nM T02226 C4USA7 44563089 Ki = 26 nM T02226 CYCA43 44563090 Ki = 4.3 nM T02226 CAY83X 44563091 Ki = 37 nM T02226 C02GYS 44563123 Ki = 22 nM T02226 CQ1GS6 44563124 Ki = 31 nM T02226 C7RF8D 44563125 Ki = 36 nM T02226 CX10VW 44563126 Ki = 13 nM T02226 C8NI7J 44563160 Ki = 9.6 nM T02226 CP9KF1 44563161 Ki = 7.1 nM T02226 CE68LK 44563162 Ki = 4.7 nM T02226 C4XLF1 44563200 Ki = 2.2 nM T02226 CBN70V 44570375 Ki = 230 nM T02226 CN08BL 44570421 Ki = 2700 nM T02226 C8WAM1 44570422 Ki = 34 nM T02226 CU79ER 44570461 Ki = 130 nM T02226 CO7Q6R 44570462 Ki = 2600 nM T02226 CF5U3J 44570463 Ki = 520 nM T02226 CV07RL 44570498 IC50 = 10 nM T02226 CS0P9O 44570499 Ki = 13 nM T02226 CN82WG 44570536 Ki = 35 nM T02226 CKN09A 44570578 Ki = 2.3 nM T02226 C3P8KA 44570579 Ki = 0.61 nM T02226 C9U7GK 44570580 Ki = 1.2 nM T02226 C0AL8Y 44570614 Ki = 0.87 nM T02226 CH4ZR3 44570615 Ki = 1.7 nM T02226 CUT6X5 44570616 Ki = 0.21 nM T02226 C38SLX 44583379 IC50 = 0.18 nM T02226 CRJ69Y 44593445 Ki = 1.7 nM T02226 CVKF91 44593545 Ki = 0.23 nM T02226 CH32KB 45267476 Ki = 0.12 nM T02226 C6BC5R 45267481 Ki = 0.28 nM T02226 C9CFX4 45269221 Ki = 2.2 nM T02226 C2S5JO 45271740 Ki = 1.4 nM T02226 CPUN79 45271754 Ki = 1.1 nM T02226 CBCA26 45273525 Ki = 9.7 nM T02226 CIPX17 45485590 Ki = 45 nM T02226 CI10RQ 45485600 Ki = 23 nM T02226 CDP21J 45485605 Ki = 0.13 nM T02226 CPVU61 45485609 Ki = 25 nM T02226 C6IG2K 45485621 Ki = 800 nM T02226 C58VXQ 45485625 Ki = 1.9 nM T02226 CF7Y8H 45485631 Ki = 14 nM T02226 CMI83V 45485640 Ki = 0.55 nM T02226 CP87FU 45485645 Ki = 1.6 nM T02226 CLJF04 45485646 Ki = 1.2 nM T02226 CQE7Z0 45485654 Ki = 3.7 nM T02226 C5J4CW 45485664 Ki = 1.8 nM T02226 C63VLU 45485665 Ki = 7.9 nM T02226 C7VRC1 45485666 Ki = 4.4 nM T02226 CK8Q9R 45485676 Ki = 56 nM T02226 C7SX0U 45485677 Ki = 0.83 nM T02226 C4UB6E 45485687 Ki = 0.26 nM T02226 CQ15ET 45485692 Ki = 0.035 nM T02226 C9LD8A 45487016 Ki = 340 nM T02226 C5AOW0 45487023 Ki = 100 nM T02226 C7HR0U 45487036 Ki = 6.6 nM T02226 CP1W4J 45487037 Ki = 240 nM T02226 C3VJ7P 45487042 Ki = 390 nM T02226 CT5I7G 45487055 Ki = 510 nM T02226 CSL40Y 45487056 Ki = 8900 nM T02226 C5W8NO 45487057 Ki = 41 nM T02226 CQZ4W1 45487059 Ki = 140 nM T02226 CP0A1T 45487060 Ki = 5000 nM T02226 CI9H4P 45487061 Ki = 66 nM T02226 C9AR7C 46174937 Ki = 0.07 nM T02226 C8KSD1 46178835 Ki = 0.3 nM T02226 CK50TO 46232527 Ki = 2511.89 nM T02226 CMFC17 46232562 Ki = 199.53 nM T02226 CCI28M 46232563 Ki = 501.19 nM T02226 C9R2OQ 46232564 Ki = 316.23 nM T02226 CH36RD 46232565 Ki = 1000 nM T02226 CBMT46 46232591 Ki = 158.49 nM T02226 CA0PE5 46232592 Ki = 794.33 nM T02226 C0N4WY 46232593 Ki = 251.19 nM T02226 C7PY3O 46232693 Ki = 199.53 nM T02226 C63ELO 46232777 Ki = 5.012 nM T02226 CPZV08 46232822 Ki = 12.59 nM T02226 C7C6EX 46884946 Ki = 55 nM T02226 C7ZI3U 46884947 Ki = 720 nM T02226 CBD92Q 46884948 Ki = 320 nM T02226 CEKT29 46884999 Ki = 6000 nM T02226 C4QT8V 46885132 Ki = 17 nM T02226 CMIO63 46885133 Ki = 8.9 nM T02226 CW0JG8 46885134 Ki = 1.4 nM T02226 CCHY85 46885135 Ki = 0.3 nM T02226 CX9A1S 46885183 Ki = 0.023 nM T02226 CS52PG 46885184 Ki = 3 nM T02226 CYFJ59 46885185 Ki = 0.41 nM T02226 CDI07R 46885186 Ki = 1.5 nM T02226 CPG38Y 46885242 Ki = 0.55 nM T02226 C8ZGX3 46885243 Ki = 0.52 nM T02226 C6H4GB 46885244 Ki = 0.12 nM T02226 CZJT73 46885245 Ki = 1.3 nM T02226 CPF6D7 46885299 Ki = 0.072 nM T02226 CK63RE 50939479 Ki = 0.046 nM T02226 C5FO7A 50939608 Ki = 0.056 nM T02226 CGSI36 51357585 Ki = 0.081 nM T02226 CJ41BC 51357854 Ki = 4.3 nM T02226 C13CSY 51357855 Ki = 0.67 nM T02226 CC9HW6 51357856 Ki = 0.066 nM T02226 CKPG40 52940673 Ki = 0.037 nM T02226 CTG24I 52940932 Ki = 0.1 nM T02226 CI1CG2 52941862 Ki = 0.11 nM T02226 CJ3AL6 52942173 Ki = 0.12 nM T02226 CY5CR0 52943413 Ki = 0.69 nM T02226 C5QHP1 52944286 Ki = 0.15 nM T02226 CK0Z5Y 52945887 Ki = 12 nM T02226 CBV64H 52947106 Ki = 1.3 nM T02226 C8C5TS 52949562 Ki = 2.2 nM T02226 CHW8L0 54580803 Ki = 0.14 nM T02226 C2FN4O 54580838 Ki = 0.38 nM T02226 C42KGV 54581838 Ki = 2.2 nM T02226 C1OEW2 54581897 Ki = 0.62 nM T02226 C5W4RL 54581909 Ki = 0.14 nM T02226 CW0HC2 54581910 Ki = 0.036 nM T02226 CLI5N2 54582783 Ki = 1 nM T02226 CR3W8B 54582784 Ki = 5.7 nM T02226 CC0WH5 54583774 Ki = 2.5 nM T02226 C4YE3A 54583775 Ki = 2.8 nM T02226 CWQ19D 54583842 Ki = 0.19 nM T02226 CE8XW4 54583843 Ki = 0.05 nM T02226 CWK2I8 54583844 Ki = 0.16 nM T02226 CH9B7I 54584803 Ki = 0.48 nM T02226 C5BF0V 54585731 Ki = 0.04 nM T02226 C0KVY7 54586710 Ki = 0.4 nM T02226 C8QSR1 54586725 Ki = 0.039 nM T02226 CD6XM5 54587752 Ki = 0.61 nM T02226 C8J7YX 54587762 Ki = 0.29 nM T02226 C1IY0P 56944164 Ki = 0.052 nM T02226 C1HYU6 57404496 Ki = 0.071 nM T02226 C1RT4K 57404529 IC50 = 0.064 nM T02226 C5EH8O 57404534 IC50 = 0.2 nM T02226 CC7N4O 57404535 IC50 = 0.019 nM T02226 CGC3T2 57794685 IC50 = 0.77 nM T02226 CXJQ07 57977594 Ki = 0.022 nM T02226 CED2Y9 57977652 Ki = 0.04 nM T02226 C8IWF0 58864250 IC50 = 98 nM T02226 C7F2PL 58864267 IC50 = 100 nM T02226 CDZU21 58864272 IC50 = 700 nM T02226 CY81QW 58864279 IC50 = 1400 nM T02226 CQ4M0I 58864296 IC50 = 36 nM T02226 C6AY0Z 58864297 Ki = 0.048 nM T02226 C05JZT 58864325 IC50 = 80 nM T02226 CZ4QL7 58864368 IC50 = 97 nM T02226 C3DR7Z 58864407 IC50 = 280 nM T02226 C3JQ0W 58864421 IC50 = 73 nM T02226 C41JYE 58864453 IC50 = 130 nM T02226 CN2D3I 58864463 IC50 = 590 nM T02226 C80MGA 58864477 IC50 = 430 nM T02226 CC68UX 58864479 IC50 = 180 nM T02226 CZU98O 58864506 IC50 = 45 nM T02226 C3EM2R 58864520 IC50 = 4500 nM T02226 C3A6HC 58901616 IC50 = 170 nM T02226 CCUA34 59554855 Ki = 64 nM T02226 C1YVE4 59554856 Ki = 0.1 nM T02226 C3EY2M 59554857 Ki = 1880 nM T02226 C0Q8JI 59554867 Ki = 115 nM T02226 C0S5YQ 59554876 Ki = 303 nM T02226 CZ8SB6 59554885 Ki = 40 nM T02226 CK96TS 59554895 Ki = 0.5 nM T02226 C8EAB3 59554924 Ki = 56 nM T02226 CJ87WH 59554934 Ki = 14 nM T02226 CZB69P 59554936 Ki = 18 nM T02226 C75RQS 59554942 Ki = 260 nM T02226 CTKE18 59554947 Ki = 1800 nM T02226 CLY1Q5 59554953 Ki = 54 nM T02226 CKP8E2 59554975 Ki = 8 nM T02226 C36LQX 59554982 Ki = 32 nM T02226 CM7W1X 59554993 Ki = 1 nM T02226 CJF23X 59555008 Ki = 118 nM T02226 C7PKE1 59555012 Ki = 7 nM T02226 CO83KR 59555024 Ki = 68 nM T02226 C3X4RA 59555031 Ki = 0.07 nM T02226 C2S4GJ 59555036 Ki = 3 nM T02226 CVS38C 59555048 Ki = 0.9 nM T02226 C3P8VH 59555055 Ki = 14 nM T02226 CL36VD 59555056 Ki = 124 nM T02226 C0WM7K 59555066 Ki = 1 nM T02226 CJH3B1 59555074 Ki = 2 nM T02226 C9OWC3 59555100 Ki = 20 nM T02226 C57IML 59555102 Ki = 203 nM T02226 CBA7R3 59555111 Ki = 865 nM T02226 CECH35 59555152 Ki = 59 nM T02226 C0O6KE 59555157 Ki = 2 nM T02226 C62BDC 59555187 Ki = 0.02 nM T02226 CD63KR 59555230 Ki = 22 nM T02226 CK8VN2 59555236 Ki = 806 nM T02226 CE1HT0 59555245 Ki = 202 nM T02226 CFI6Z8 59555258 Ki = 10 nM T02226 CO4VJ9 59555260 Ki = 52 nM T02226 C51OYL 59555274 Ki = 763 nM T02226 C42QTA 59555277 Ki = 30 nM T02226 CA9GL6 59555326 Ki = 45 nM T02226 COJ84D 59555331 Ki = 2 nM T02226 CV13OQ 62705051 EC50 = 3 nM T02226 C4YHM2 68857312 EC50 = 0.15 nM T02226 C0GH3B 69747490 Ki = 0.11 nM T02226 CUQ78F 70681261 IC50 = 380 nM T02226 CS0P8G 70681269 IC50 = 220 nM T02226 CD4W6J 70681270 IC50 = 0.12 nM T02226 CA0GP3 70681361 IC50 = 0.1 nM T02226 C83WEP 70681362 IC50 = 0.24 nM T02226 CNA09E 70682193 Ki = 7.2 nM T02226 C9S1RD 70682194 Ki = 250 nM T02226 C78DAT 70683458 IC50 = 3 nM T02226 CPS24M 70683493 IC50 = 0.093 nM T02226 CP09GW 70684297 Ki = 750 nM T02226 CU3F7D 70684299 IC50 = 210 nM T02226 C2GH6T 70685453 IC50 = 32 nM T02226 C4MIR9 70685454 IC50 = 120 nM T02226 CXK7N2 70685565 IC50 = 0.33 nM T02226 CT8CJ5 70685566 IC50 = 0.39 nM T02226 C4F2XL 70685594 IC50 = 6.8 nM T02226 C5Z4TE 70685595 IC50 = 0.28 nM T02226 CUO9N4 70686450 Ki > 1000 nM T02226 C92GRS 70686451 Ki = 1900 nM T02226 CY3F6J 70686453 IC50 = 330 nM T02226 CDZ9Y3 70686454 IC50 = 8500 nM T02226 C4DP6B 70687597 IC50 = 0.049 nM T02226 C06YZS 70687709 IC50 = 4.4 nM T02226 CT6I9A 70687746 IC50 = 6.6 nM T02226 C1VI4M 70688551 Ki > 1000 nM T02226 CL4I8H 70688552 Ki = 2.5 nM T02226 CMJ9P6 70688553 Ki > 1000 nM T02226 COF79Z 70688557 IC50 = 4 nM T02226 CW1U7R 70689654 IC50 = 11 nM T02226 CL2PV7 70689756 IC50 = 0.27 nM T02226 C58NQB 70690613 Ki = 300 nM T02226 C80HOI 70690614 Ki = 1400 nM T02226 C0YA3Z 70690615 Ki = 0.65 nM T02226 CFQ7Z0 70690616 Ki = 16 nM T02226 C4BG7D 70690617 Ki = 250 nM T02226 C8H0NL 70690619 IC50 = 170 nM T02226 C86BMI 70691910 IC50 = 0.33 nM T02226 CND85T 70692757 Ki = 2100 nM T02226 CF1D0A 70692758 Ki > 1000 nM T02226 CRDT90 70692759 Ki = 230 nM T02226 CF4R5I 70692761 IC50 = 860 nM T02226 CKN87D 70693851 IC50 = 99 nM T02226 C5ZC4H 70693987 IC50 = 1.9 nM T02226 COP8L5 70694798 Ki > 1000 nM T02226 CVH1E7 70694802 Ki = 0.55 nM T02226 CV6LI0 70694803 EC50 = 15 nM T02226 C1P7ZJ 70694804 EC50 = 13 nM T02226 C0UPX1 70694861 Ki = 940 nM T02226 CWSV01 70695973 IC50 = 890 nM T02226 CL89KS 70695974 IC50 = 4.6 nM T02226 CP91SM 70696075 IC50 = 0.1 nM T02226 C2LP3E 70696076 IC50 = 12 nM T02226 C5S7CI 70696077 IC50 = 0.24 nM T02226 CSG16Y 70696078 IC50 = 1.2 nM T02226 CDPJ35 70696079 IC50 = 0.042 nM T02226 CBDN32 70696080 IC50 = 1.3 nM T02226 CK42BQ 70696845 Ki = 2400 nM T02226 C62EGB 70696847 Ki = 84 nM T02226 CH4U7X 70696851 IC50 = 1400 nM T02226 CZ4SR9 71569374 Ki = 27 nM T02226 CS2VA3 71569375 Ki = 0.032 nM T02226 C3OM9G 71569532 Ki = 11 nM T02226 C9WNA4 71569533 Ki = 0.015 nM T02226 C6TI0G 72190777 IC50 = 0.39 nM T02226 C85DFY 72190778 IC50 = 0.37 nM T02226 CE8OT0 72191391 IC50 = 0.22 nM T02226 CYO9R8 72191392 IC50 = 0.26 nM T02226 C9VUN4 72191699 IC50 = 2.9 nM T02226 C7Y8BN 73346897 IC50 = 3 nM T02226 CQ58KP 73347057 IC50 = 910 nM T02226 C85OLV 73348402 IC50 = 8 nM T02226 C7JX6P 73348426 IC50 = 14 nM T02226 CS34XQ 73351480 IC50 = 21.9 nM T02226 CJ46SV 73352727 IC50 = 2 nM T02226 C1WD2P 73352946 IC50 = 9 nM T02226 CWS2T8 73352948 Ki = 0.028 nM T02226 CJH08Z 73353203 IC50 = 3548.13 nM T02226 CT7R5K 73355345 IC50 = 1.7 nM T02226 C4G0TL 73356026 IC50 = 11.2 nM T02226 CP7Y1K 73356029 IC50 = 0.5 nM T02226 C0O5XH 73356030 IC50 = 20.2 nM T02226 C6Q2RG 73356952 Ki = 0.017 nM T02226 CHTC49 76310534 Ki = 9 nM T02226 CSUE07 76310551 Ki = 282 nM T02226 C31NWZ 76321477 Ki = 0.03 nM T02226 C7FVX4 76325057 Ki = 297 nM T02226 CSE87P 76332330 Ki = 1 nM T02226 CXB49M 86298538 EC50 = 100 nM T02226 CH2D9L 86298539 IC50 = 25 nM T02226 CTV8B0 118718879 IC50 = 19000 nM T02226 CDLX50 134130160 IC50 = 0.032 nM T02226 CXHY05 135461116 Ki = 26 nM T02226 CHS46O 46905052 Ki = 0.23 nM T02226 D02NMK 44274034 IC50 = 159 nM T02226 D05LMD 16134896 IC50 = 0.5 nM T02226 D05MSG 44593666 Ki = 0.0128 nM T02226 D08GZJ 54580850 Ki = 0.05 nM T02226 D09TDY 23582940 Ki = 0.35 nM T02226 D0B8HD 44274033 IC50 = 29 nM T30823 D00FGR 3599 IC50 = 25000 nM T30823 D03GET 4055 IC50 = 6900 nM T30823 D0H4JM 8969 IC50 = 22300 nM T30823 D02UOE 160142 IC50 > 20 ug.mL-1 T30823 CAD58I 2876 IC50 = 4500 nM T30823 CF1MI3 3136 IC50 = 8900 nM T30823 CI9TK0 3884 IC50 = 33200 nM T30823 C3PIF6 21076 IC50 = 12000000 nM T30823 C8JV3A 24465 IC50 = 30000 nM T30823 C6G5AH 79441 IC50 = 22300 nM T30823 C3GIJ7 97529 IC50 = 45300 nM T30823 CFS1T8 133223 IC50 = 110000 nM T30823 CXJ37I 231852 Ki = 2300 nM T30823 CK6M9P 233507 IC50 = 15400 nM T30823 C0UXN2 236650 IC50 = 45700 nM T30823 C7HSE4 237492 IC50 = 36000 nM T30823 C0O2FK 259836 IC50 = 5500 nM T30823 C7H4JI 268982 IC50 = 86000 nM T30823 CZA6G5 274127 Ki = 70 nM T30823 CV6AX0 320851 IC50 = 1500 nM T30823 C05EMO 351827 IC50 = 2300 nM T30823 C75COU 470952 IC50 = 2400 nM T30823 CO4J7N 470958 IC50 = 32900 nM T30823 CH35LS 662869 IC50 = 13000 nM T30823 CDI2W3 719031 IC50 = 20300 nM T30823 C2B6EK 752982 IC50 = 25700 nM T30823 C5MQP8 852158 IC50 = 17800 nM T30823 C6OSR1 914570 IC50 = 5500 nM T30823 CI87JW 1001784 IC50 = 7500 nM T30823 C9K1SE 1177946 IC50 = 17200 nM T30823 CFR61E 1307198 IC50 = 12300 nM T30823 CQW6F7 1308005 IC50 = 20100 nM T30823 C9VW4Y 1332846 IC50 = 19000 nM T30823 CKD92S 1383304 IC50 = 800 nM T30823 C3VIK9 1398345 IC50 = 3280 nM T30823 C91NQB 1400320 IC50 = 7100 nM T30823 CSC9W6 1400627 IC50 = 6000 nM T30823 CH3M0Z 1401217 IC50 = 9200 nM T30823 C4U8DM 1413573 IC50 = 11500 nM T30823 C8J2ZI 1864385 IC50 = 11100 nM T30823 C7M4ID 1895639 IC50 = 5000 nM T30823 CU0A3X 1921859 IC50 = 2900 nM T30823 C9CS3K 1925936 IC50 = 8200 nM T30823 C4RH2W 1933357 IC50 = 2100 nM T30823 CRFK64 1953519 IC50 = 13300 nM T30823 C9JQ2O 1968455 IC50 = 13100 nM T30823 CO9ST2 2446135 IC50 = 13000 nM T30823 COE91V 2742421 IC50 = 12200 nM T30823 C7JO4Q 2820003 IC50 = 2700 nM T30823 C5AZL4 2941397 IC50 = 17800 nM T30823 CYN3Z9 4263321 IC50 = 2300 nM T30823 C6R3WL 4343361 IC50 = 6300 nM T30823 CWIC65 5279637 IC50 = 5400 nM T30823 C8CTS9 5279656 IC50 = 50 nM T30823 C0PCZ3 5932584 IC50 = 2800 nM T30823 CU65JT 5998084 IC50 = 3400 nM T30823 C14LAC 6161281 IC50 = 2400 nM T30823 CR6O8V 6166563 IC50 > 10000 nM T30823 CYI5R1 6274486 IC50 = 3400 nM T30823 C4VM8J 9173830 IC50 = 10200 nM T30823 CP3AO9 9356353 IC50 = 6500 nM T30823 CZ93IR 9356454 IC50 = 4000 nM T30823 CF79QB 9421427 IC50 = 9500 nM T30823 C1DMN7 9850223 IC50 = 7800 nM T30823 CIAT52 9865848 IC50 = 15000 nM T30823 C3MUO6 9903359 IC50 = 5700 nM T30823 C0CJ7U 9926573 IC50 = 5500 nM T30823 CRU8E0 9978702 IC50 = 890 nM T30823 COU6V1 9978703 IC50 = 860 nM T30823 CA75NG 9985013 IC50 = 163000 nM T30823 COB58D 10092773 IC50 = 440 nM T30823 C3A8JL 10256983 IC50 = 30000 nM T30823 CUD28W 10318951 IC50 = 13000 nM T30823 C2B8AM 10476452 IC50 = 480 nM T30823 CI48ME 10507182 IC50 > 100000 nM T30823 CT38OX 10531514 IC50 > 100000 nM T30823 C0ZTJ9 10572551 IC50 > 1000000 nM T30823 CCUH28 10573797 IC50 = 24200 nM T30823 CJ69GO 10598282 IC50 = 290000 nM T30823 CQO97K 10621802 IC50 = 2200 nM T30823 CAIE64 10647004 IC50 = 10500 nM T30823 C5O4HY 10647065 IC50 = 700 nM T30823 C0IMZ1 10669449 IC50 > 50000 nM T30823 C8A3EI 10671123 IC50 = 460000 nM T30823 CX6YO3 10693079 IC50 = 13300 nM T30823 CXL14P 10695263 IC50 = 2900 nM T30823 C5TQ8B 10716686 IC50 = 9700 nM T30823 C2MRA7 10716972 IC50 = 490000 nM T30823 CDR2X1 10745262 IC50 > 100000 nM T30823 CE2FZ5 10763151 IC50 = 500000 nM T30823 CP94UD 10765299 IC50 = 5100 nM T30823 CVY0K4 10768361 IC50 = 900 nM T30823 CNE54S 10793410 IC50 > 100000 nM T30823 C0O5ZF 10811706 IC50 = 36300 nM T30823 CDRL67 10835677 IC50 = 2400 nM T30823 CU9V1B 10837228 IC50 = 40000 nM T30823 C9WQA1 10839788 IC50 = 2100 nM T30823 CTY50V 10883523 IC50 = 890 nM T30823 CT4H0O 11006141 IC50 = 163000 nM T30823 C5A3WY 11200445 IC50 = 1000 nM T30823 CXN1S5 11269661 IC50 = 9400 nM T30823 CQJ07W 11299775 IC50 > 100000 nM T30823 CU4E2B 11391905 IC50 > 100000 nM T30823 CRPL64 11516963 IC50 = 73300 nM T30823 C8V9FL 11678073 IC50 = 70700 nM T30823 CV6K2W 11796020 IC50 = 29000 nM T30823 CM1XL8 11844603 IC50 > 100000 nM T30823 C75UVA 11844604 IC50 > 100000 nM T30823 CG8ZU9 12020703 IC50 = 5800 nM T30823 CHPQ20 12020709 IC50 = 5900 nM T30823 CD3K8H 12387018 IC50 = 26100 nM T30823 CP8FX1 12824032 IC50 = 11600 nM T30823 CG18HV 13690444 IC50 = 1000000 nM T30823 CSC25V 14149682 IC50 = 44400 nM T30823 CY3JU7 14646108 IC50 > 100000 nM T30823 C8SQZ0 15549018 IC50 = 990000 nM T30823 C50VIT 15673044 IC50 = 9500 nM T30823 CU8J6A 16126459 IC50 = 4700 nM T30823 C8CSM3 16126550 IC50 = 8100 nM T30823 C29ZMK 16126551 IC50 = 6300 nM T30823 C3TPL7 16126552 IC50 = 5100 nM T30823 C4Z6BF 17483715 IC50 = 2400 nM T30823 C04GYC 17531735 IC50 = 5600 nM T30823 CX42CP 17554676 IC50 = 6400 nM T30823 CFU3D7 18350018 IC50 = 5100 nM T30823 C5O0SV 24204784 Ki = 1700 nM T30823 C3P6HS 24857863 IC50 = 2600 nM T30823 CT5AV2 25147777 IC50 = 4070 nM T30823 C6NR5D 44249868 IC50 = 4700 nM T30823 C2TV9N 44303254 IC50 > 360000 nM T30823 CK78HD 44303432 IC50 = 6300 nM T30823 C1X8YT 44303433 IC50 = 74000 nM T30823 CPC2M1 44303451 IC50 = 29000 nM T30823 CZ5MD3 44303453 IC50 = 31000 nM T30823 CT2HK6 44303463 IC50 = 32000 nM T30823 CN89QP 44303489 IC50 > 100000 nM T30823 C7E4AP 44303513 IC50 = 2800 nM T30823 C5H0VL 44303516 IC50 = 170000 nM T30823 C5Y6QE 44303518 IC50 > 100000 nM T30823 C7GJ6P 44303523 IC50 = 60000 nM T30823 CHK98F 44303528 IC50 = 10600 nM T30823 CBI8O6 44303580 IC50 = 46300 nM T30823 C0X8JR 44303638 IC50 > 310000 nM T30823 CXN80T 44303639 IC50 > 290000 nM T30823 CZTE47 44303667 IC50 = 3800 nM T30823 CYL2E5 44303668 IC50 = 8400 nM T30823 CIT1K3 44303684 IC50 > 100000 nM T30823 CMPA04 44303685 IC50 > 100000 nM T30823 C7YN6L 44318744 IC50 > 50000 nM T30823 C1O5XM 44319185 IC50 = 21000000 nM T30823 CK69BS 44320206 IC50 = 15000 nM T30823 CD9Z6B 44320207 IC50 > 300000 nM T30823 CWH8Z1 44321838 IC50 = 100000 nM T30823 CMD5V4 44321840 IC50 = 300000 nM T30823 CSB0Y5 44322128 IC50 = 1000000 nM T30823 CF7T3B 44322130 IC50 = 380000 nM T30823 C2PI0F 44322155 IC50 = 610000 nM T30823 CTN35X 44361793 IC50 = 4000 nM T30823 CF3UO8 44371035 IC50 > 300000 nM T30823 CK2Q1T 44371036 IC50 = 32000 nM T30823 C3MVG1 44371682 IC50 = 9000 nM T30823 C93XSD 44371683 IC50 = 94000 nM T30823 CT2S0H 44371696 IC50 > 300000 nM T30823 CLH29B 44380956 IC50 = 11700 nM T30823 CWZ2G9 44381072 IC50 = 1900 nM T30823 CVF24B 44381278 IC50 = 9300 nM T30823 CE6PU8 44381470 IC50 = 7800 nM T30823 CFL91W 44392831 IC50 = 3900 nM T30823 C54CFD 44392873 IC50 = 8200 nM T30823 CKO5A0 44405932 IC50 > 100000 nM T30823 C4JZ1E 44405933 IC50 > 100000 nM T30823 CBX34H 44405951 IC50 > 100000 nM T30823 CAJ5T4 44405958 IC50 > 100000 nM T30823 CSLQ50 44405959 IC50 > 100000 nM T30823 C0Q5NW 44406035 IC50 = 69200 nM T30823 CX28MD 44406938 IC50 = 1330 nM T30823 C4VO7S 44407055 IC50 = 10000 nM T30823 CYW68I 44409605 IC50 = 12750 nM T30823 CGX23J 44409674 IC50 = 20310 nM T30823 CTM56S 44409675 IC50 = 5430 nM T30823 C6E4UN 44409680 IC50 = 22060 nM T30823 C25MUW 44409681 IC50 = 3960 nM T30823 CTL17C 44409833 IC50 = 21870 nM T30823 CB31QM 44409834 IC50 = 8810 nM T30823 CY6QB9 44409856 IC50 = 5960 nM T30823 C23ERY 44409919 IC50 = 6870 nM T30823 CB96NM 44409921 IC50 = 27580 nM T30823 C56DNZ 44409999 IC50 = 3970 nM T30823 CH08EI 44410004 IC50 = 11820 nM T30823 C94QYM 44410005 IC50 = 4900 nM T30823 CJUM36 44415112 IC50 > 100000 nM T30823 C0S8RA 44424744 IC50 = 44300 nM T30823 C9SJ3O 44424745 IC50 = 4500 nM T30823 C7ZIL9 44576906 IC50 > 100000 nM T30823 CVH40K 44576907 IC50 = 78000 nM T30823 CA6U8V 44576948 IC50 = 1900 nM T30823 CL3N5K 44576949 IC50 > 100000 nM T30823 CIPX63 44576971 IC50 > 100000 nM T30823 C3ZQ0C 44576972 IC50 > 100000 nM T30823 CDN1K3 44576973 IC50 = 39000 nM T30823 C4XG6B 44576975 IC50 = 2900 nM T30823 CT9VE2 44576976 IC50 = 1700 nM T30823 CJ5SN3 44577007 IC50 = 1600 nM T30823 CW26GM 44577008 IC50 = 37000 nM T30823 CGCE54 44577009 IC50 = 50000 nM T30823 CLIK47 45267539 IC50 = 7100 nM T30823 C3IQM0 45267545 IC50 = 14500 nM T30823 C2MDQ6 45270955 IC50 = 11400 nM T30823 CCG19S 45922965 IC50 = 30700 nM T30823 C7ZS4V 46218884 IC50 = 26000 nM T30823 CE4PU6 46873799 IC50 = 27000 nM T30823 C9FW7G 46946067 IC50 = 28000 nM T30823 C6QCU0 52942665 IC50 = 78000 nM T30823 C73QHN 52943900 IC50 = 62000 nM T30823 CB4U2R 52945119 IC50 = 96000 nM T30823 CG3TM0 52948739 IC50 = 70000 nM T30823 CIE87V 54585167 IC50 = 440 nM T30823 CE94WN 54587113 IC50 = 2000 nM T30823 CAEU25 54587114 IC50 = 5100 nM T30823 CJV2M8 54587115 IC50 = 800 nM T30823 CHM5V3 56660070 IC50 > 120000 nM T30823 CHOF39 56670422 IC50 = 26800 nM T30823 CL3N0K 56673907 IC50 = 118700 nM T30823 CAL96I 56673908 IC50 = 53000 nM T30823 CEK3S2 56680547 IC50 > 120000 nM T30823 CN3EW7 56683882 IC50 > 120000 nM T30823 C5CQY2 56683883 IC50 = 51600 nM T30823 CV4PW2 56683884 IC50 = 24300 nM T30823 CWBE16 66525293 IC50 = 36400 nM T30823 CTQ95V 71461600 IC50 = 36300 nM T30823 CJ2ZQ7 71697056 IC50 = 5800 nM T30823 C6PFD1 73345215 IC50 = 8500 nM T30823 CGC60U 73346748 IC50 = 5500 nM T30823 CHBJ65 73346749 IC50 = 5500 nM T30823 C5DV3I 73346750 IC50 = 900 nM T30823 C5PYT7 73349825 IC50 = 22700 nM T30823 C3QPK5 73349826 IC50 = 6900 nM T30823 C3WGM7 73351344 IC50 = 700 nM T30823 C15NCG 73354312 IC50 = 24500 nM T30823 CS76KU 90666197 IC50 = 2200 nM T30823 C96RMI 90666198 IC50 = 6900 nM T30823 C1Y9EK 90666199 IC50 = 17500 nM T30823 CZ50TY 90666200 IC50 = 25000 nM T30823 CM92PW 121344571 IC50 <= 9000 nM T30823 CRFQ07 124165614 Ki = 600 nM T30823 C6DCR0 135420883 IC50 = 12600 nM T30823 CBD5C3 135420929 IC50 = 12700 nM T30823 CS1KZ3 135441149 IC50 = 6700 nM T30823 C0P6TV 135444298 IC50 = 9100 nM T30823 CG2Q6N 135444322 IC50 = 14300 nM T30823 C9NYV1 135444837 IC50 = 30700 nM T30823 CRV42A 135451647 IC50 = 6200 nM T30823 C2I3NM 135458252 IC50 = 4100 nM T30823 CX9AV5 135469884 IC50 = 4270 nM T30823 C04TVF 135512954 IC50 = 10100 nM T30823 CV1ZB2 135522709 IC50 = 7800 nM T30823 C78BVZ 135527488 IC50 = 7700 nM T30823 CJRX49 135529547 IC50 = 11100 nM T30823 CF8V7A 135529575 IC50 = 15400 nM T30823 CDP6X2 135629644 IC50 = 5100 nM T30823 CCMG69 135658050 IC50 = 8100 nM T30823 CO06BL 135665679 IC50 = 12800 nM T30823 CSC48W 135700427 IC50 = 10300 nM T30823 C2V7NL 135797380 IC50 = 11400 nM T30823 C27EYJ 135797381 IC50 = 15400 nM T30823 CZOL36 135797386 IC50 = 12700 nM T30823 CBX75S 135797387 IC50 > 100000 nM T30823 C2L6UZ 135797388 IC50 = 7350 nM T30823 C0S1VO 135797389 IC50 = 10200 nM T30823 CS40TI 135797392 IC50 > 100000 nM T30823 C0RJW6 135797397 IC50 = 6860 nM T30823 C5UL0V 135955126 IC50 = 7040 nM T30823 C9YRO4 135966042 IC50 = 17300 nM T30823 C85VGD 136069445 IC50 = 5550 nM T30823 CQ7L2H 136254273 IC50 = 6250 nM T30823 C5C1XF 136254274 IC50 = 10700 nM T30823 CL4A5E 136254275 IC50 = 11700 nM T30823 CH7N3Z 136254276 IC50 = 8670 nM T30823 CL4ZM7 136254277 IC50 = 12300 nM T30823 CAHC90 136254278 IC50 = 12600 nM T30823 CQ84LN 136254279 IC50 = 19000 nM T30823 CBEU97 136254280 IC50 = 8500 nM T30823 C3LK1C 136254281 IC50 = 6220 nM T30823 CXZ40A 137228141 Ki = 3100 nM T30823 C4Y2TB 137228142 IC50 = 8300 nM T30823 C13DWG 137228143 IC50 = 7800 nM T30823 C15MJN 137228144 IC50 = 7300 nM T30823 C3AY7U 137631699 IC50 = 1200 nM T30823 COA4K6 137632835 IC50 = 2880 nM T30823 C9A6MY 137632994 IC50 = 2850 nM T30823 C2MTQ4 137633618 IC50 = 4330 nM T30823 C2K0GE 137636105 IC50 = 2190 nM T30823 CL1HE3 137641758 IC50 = 6600 nM T30823 C28DUQ 137642390 IC50 = 27460 nM T30823 CO71IL 137643613 IC50 = 13000 nM T30823 C30XET 137646265 IC50 = 4040 nM T30823 CKU6O7 137648500 IC50 = 3500 nM T30823 C5DKW8 137650422 IC50 = 2570 nM T30823 C15EWQ 137653741 IC50 = 1500 nM T30823 C4E9QK 137654526 IC50 = 3370 nM T30823 CQW02T 137656106 IC50 = 2900 nM T30823 CU9E1R 137656483 IC50 = 3110 nM T30823 CD2JY1 137658569 IC50 = 7730 nM T30823 CWE7I3 137659432 IC50 = 3230 nM T30823 CVO34Q 137659449 IC50 = 1610 nM T30823 CNMJ89 138911333 Ki = 3000 nM T30823 CB2D3K 139600304 IC50 = 530 nM T30823 CIN0D1 145964209 IC50 = 14100 nM T30823 CA7G2L 145966685 IC50 = 20500 nM T30823 C7EQ9U 145978118 IC50 = 11400 nM T30823 CW36SM 145978264 IC50 = 32900 nM T30823 C8V0XS 155512987 Ki = 600 nM T30823 CCQ48F 155531806 IC50 = 1200 nM T30823 C4D5MV 155543902 IC50 = 540 nM T30823 D00ANJ 1897797 IC50 = 15000 nM T30823 D00SAA 14828129 IC50 = 11180 nM T30823 D04OXY 16871 IC50 = 2300 nM T30823 D07JRA 44409685 IC50 = 7830 nM T30823 D08GWQ 44409669 IC50 = 5860 nM T30823 D0CJ6P 44577010 IC50 = 8000 nM T30823 D0GE3O 44576946 IC50 = 13000 nM T30823 D0J1KH 262093 IC50 = 1400 nM T30823 D0N7YT 44409922 IC50 = 7060 nM T30823 D0P0IE 10205 IC50 = 700 nM T30823 D0W1SP 44576974 IC50 = 12000 nM T30823 D0X5WD 44409841 IC50 = 10880 nM T00176 D07XSN 6253 IC50 = 20 nM T00176 D0E7PQ 5311 Ki > 20000 nM T00176 D0H6QU 6005 IC50 = 195 nM T00176 D01KTG 71678098 Ki = 0.21 nM T00176 D03YSQ 53476877 Ki = 0.88 nM T00176 D04SXL 91972012 Ki < 1 nM T00176 D08EOW 57406853 IC50 = 18 nM T00176 D0C1WR 58573469 IC50 = 0.6 nM T00176 D0OC4O 53358942 IC50 = 6 nM T00176 D0Q7AG 53240420 Ki = 1.3 nM T00176 D0Z0HH 3503 Ki > 25000 nM T00176 C6NG1O 179269 IC50 > 295000 nM T00176 CJ38BD 656933 IC50 = 420 nM T00176 CO9W5L 722626 Ki = 93 nM T00176 C3I6NZ 745150 IC50 = 4700 nM T00176 C7GY1X 869152 Ki > 25000 nM T00176 CK45IC 1036120 IC50 = 720 nM T00176 C6SBD8 1043193 IC50 = 3300 nM T00176 CN1W8P 1109690 IC50 = 110 nM T00176 C4TP0I 1109692 IC50 = 170 nM T00176 CG2LM0 1114145 IC50 > 75000 nM T00176 CV2FP8 1317466 EC50 = 840 nM T00176 CQ4XS9 1354867 IC50 = 8400 nM T00176 CMQ4E8 1732573 IC50 = 199 nM T00176 CE87OK 1883338 IC50 > 100000 nM T00176 C0V6NK 2337251 IC50 = 150 nM T00176 CWA18R 2487662 Ki = 230 nM T00176 CC74TR 2771353 Ki = 3260 nM T00176 CEYB92 3117824 IC50 = 180 nM T00176 CD0M2Z 3121559 IC50 = 300 nM T00176 C51QGW 3608080 IC50 = 74000 nM T00176 C4X0LM 5288631 IC50 = 140 nM T00176 C5VL3P 5760860 IC50 = 256 nM T00176 CN8ML2 5760862 IC50 = 230 nM T00176 C1CNQ5 5760865 IC50 = 163 nM T00176 CFAM21 6213796 Ki = 140 nM T00176 C7EOJ1 9812342 IC50 = 5 nM T00176 CAVJ32 9917797 IC50 = 394 nM T00176 C4V3UI 10008863 IC50 = 100 nM T00176 C8X9ZG 10015619 IC50 = 1700 nM T00176 C73QDP 10078330 IC50 = 140 nM T00176 CAK8E4 10124724 IC50 = 16000 nM T00176 CEFG43 10173806 IC50 = 90 nM T00176 CTP32Q 11192949 IC50 = 3600 nM T00176 CGPZ09 11351960 Ki = 8.5 nM T00176 CDAT72 11433190 Ki = 6.4 nM T00176 CZT37E 11447214 IC50 = 50 ug.mL-1 T00176 CLN93X 11475818 Ki = 8460 nM T00176 C39BQK 11502965 IC50 = 3000 nM T00176 CXLC39 11512421 Ki = 13 nM T00176 CVE4N6 11512578 Ki = 1.7 nM T00176 C84IZQ 11526064 Ki = 38 nM T00176 CD91JP 11541499 Ki = 39 nM T00176 C69KNG 11571200 IC50 = 704 nM T00176 CUK7A9 11591070 IC50 = 700 nM T00176 C9B2JR 11599265 Ki = 0.6 nM T00176 C0VBF4 11620161 Ki = 44 nM T00176 CKF7P5 11621174 Ki = 4000 nM T00176 C1GXO9 11663211 Ki = 170 nM T00176 CVM86J 11706629 IC50 = 710 nM T00176 C10CJT 11848430 IC50 = 26200 nM T00176 C2OV1A 11952735 IC50 = 787 nM T00176 CI1W4K 11952782 IC50 = 790 nM T00176 CNP1K4 11952783 IC50 = 250 nM T00176 C9GXP3 11952784 IC50 = 13100 nM T00176 CI3X7J 11952815 IC50 = 7000 nM T00176 CQ98BE 11952816 IC50 = 980 nM T00176 CQ75ON 11952817 IC50 = 1040 nM T00176 C0O8HI 11953136 IC50 = 2600 nM T00176 CDPM69 11953137 IC50 = 2700 nM T00176 CB7DS4 11953254 IC50 = 1110 nM T00176 CC0E8F 16755649 IC50 = 108 nM T00176 CG6V2A 17754546 IC50 = 30 nM T00176 CTX3P7 17754588 IC50 = 23 nM T00176 C1OYK9 17754765 IC50 = 18 nM T00176 C4CK8P 17754800 IC50 = 209 nM T00176 CVG1F6 17754801 IC50 = 22 nM T00176 CA56GZ 17754803 IC50 = 14 nM T00176 CUXR60 17754844 IC50 = 33 nM T00176 CKC2H5 17754845 IC50 = 46 nM T00176 CU8X1T 17754846 IC50 = 26 nM T00176 CXU2M0 21060006 IC50 = 6250 nM T00176 CK3O6C 21060010 IC50 = 2390 nM T00176 CS57AK 21060012 IC50 = 2700 nM T00176 CX30SL 22046756 IC50 = 2180 nM T00176 CYR54U 22046762 IC50 = 38000 nM T00176 C52XTW 22046784 IC50 = 3330 nM T00176 CGRD68 22046788 IC50 = 10200 nM T00176 C8UQA5 22046890 IC50 = 1090 nM T00176 C0VE5D 23642310 IC50 = 40 nM T00176 C4K2VR 24813118 IC50 > 60000 nM T00176 C5KD6W 24823666 IC50 = 2300 nM T00176 CF89BQ 24877503 Ki = 5 nM T00176 CMU65Q 24936079 IC50 = 11500 nM T00176 CG9AI6 24968163 IC50 = 340 nM T00176 C5Z6QL 24969086 Ki = 109 nM T00176 CLZ0R7 25001753 Ki = 12.6 nM T00176 C7S0MR 25147779 IC50 = 58600 nM T00176 CF3O6C 25227848 IC50 = 360 nM T00176 CB46WK 25227971 IC50 = 450 nM T00176 CR81DT 44176172 IC50 = 810 nM T00176 CQ68ZK 44176173 IC50 = 2440 nM T00176 C7TL4A 44176174 IC50 > 12500 nM T00176 CB25UE 44176175 IC50 = 11600 nM T00176 CR4AN8 44176176 IC50 = 3600 nM T00176 CD3Z4A 44176177 IC50 = 8600 nM T00176 CHFN54 44176178 IC50 = 25000 nM T00176 CG6M7W 44176179 IC50 = 19000 nM T00176 CT27FS 44176180 IC50 = 2830 nM T00176 C1UEP3 44176181 IC50 = 12200 nM T00176 C1DW0B 44176182 IC50 = 5410 nM T00176 C4VLD9 44176183 IC50 = 5660 nM T00176 CPB7S3 44176184 IC50 > 12500 nM T00176 C8ONC2 44176185 IC50 = 540 nM T00176 C3W5VC 44176186 IC50 = 2120 nM T00176 CB79MI 44176187 IC50 = 850 nM T00176 CX0AO9 44176188 IC50 = 31000 nM T00176 CM2PZ6 44176189 IC50 = 27000 nM T00176 C46RMP 44176199 IC50 = 13000 nM T00176 C4A9DW 44176200 IC50 = 13300 nM T00176 CW2DI4 44390543 IC50 = 1700 nM T00176 C3LVK1 44390641 IC50 = 15000 nM T00176 C8UV1S 44390659 IC50 = 30000 nM T00176 CC48NA 44390678 IC50 = 13000 nM T00176 CAT79D 44411888 IC50 = 5400 nM T00176 CX1KO7 44411911 IC50 = 1550 nM T00176 CO85XV 44412051 IC50 = 9000 nM T00176 C9C7LQ 44412055 IC50 = 2820 nM T00176 CQ06FT 44412088 IC50 = 4350 nM T00176 C6ETU0 44412108 IC50 = 2150 nM T00176 CDF75C 44412115 IC50 = 36000 nM T00176 C5KBE2 44412732 IC50 = 250 nM T00176 CV1IW3 44412775 IC50 = 850 nM T00176 CSPG43 44421706 IC50 = 13100 nM T00176 CKB3E7 44421760 IC50 > 100000 nM T00176 CMR2A1 44421777 IC50 = 19600 nM T00176 CL74BZ 44472949 IC50 > 100000 nM T00176 CMZ34J 44472950 IC50 = 85000 nM T00176 CDG73N 44472951 IC50 = 63000 nM T00176 C1CA8S 44472952 IC50 = 43000 nM T00176 C76YPC 44472953 IC50 = 18000 nM T00176 CAJ5Q2 44472954 IC50 = 20000 nM T00176 CS9TJ0 44472955 IC50 = 38000 nM T00176 C9F6EY 44472956 IC50 = 17000 nM T00176 CY9G8S 44472957 IC50 = 9200 nM T00176 CU49PM 44472958 IC50 = 24000 nM T00176 CK5U1C 44472959 IC50 = 41000 nM T00176 CA86ZW 44472960 IC50 > 100000 nM T00176 CZ4LN0 44472961 IC50 = 13000 nM T00176 C6MGL0 44472962 IC50 = 13000 nM T00176 CQ84LW 44472963 IC50 = 12000 nM T00176 CG7P3B 44472964 IC50 = 10000 nM T00176 C4CON7 44472965 IC50 = 8200 nM T00176 CPK9V3 44472966 IC50 = 6400 nM T00176 C5BYN0 44472968 IC50 = 17000 nM T00176 C3Z4SR 44472969 IC50 = 6600 nM T00176 C94UNC 44472970 IC50 = 8200 nM T00176 C6HOC3 44472971 IC50 = 2800 nM T00176 CST25L 44472972 IC50 = 2800 nM T00176 C8QNJ9 44472973 IC50 = 2600 nM T00176 CS95EF 44472974 IC50 = 2300 nM T00176 COM24Y 44472975 IC50 = 2900 nM T00176 CNOT62 44472976 IC50 = 13000 nM T00176 C4TI7C 44472977 IC50 = 5900 nM T00176 C20FAI 44549764 IC50 = 70 nM T00176 CAT3M4 44549891 IC50 = 16000 nM T00176 C5W0VC 44582364 IC50 = 10 nM T00176 CVP7N1 44588489 IC50 = 58600 nM T00176 C8SQD6 44588490 IC50 = 120800 nM T00176 C3ZRQ0 44594120 IC50 = 1900 nM T00176 CV0JR2 44595318 IC50 = 1500 nM T00176 C19NYL 44595320 IC50 = 1400 nM T00176 CW43JX 44595458 IC50 = 4700 nM T00176 C2L0EW 44595459 IC50 = 3200 nM T00176 CIYE24 44595460 IC50 = 2500 nM T00176 CO1SI7 44595461 IC50 = 3500 nM T00176 CQA0T9 44595462 IC50 = 400 nM T00176 C40UIR 44595463 IC50 = 380 nM T00176 C7RP4U 44595605 IC50 = 400 nM T00176 CSO8H7 44595606 IC50 = 660 nM T00176 CQZ20G 44596000 IC50 = 9.5 nM T00176 CNO1W8 44606480 Ki = 1.5 nM T00176 C1BEN9 44606481 Ki = 2 nM T00176 CDT95E 44606645 Ki = 0.8 nM T00176 C5ATF9 44606646 Ki = 4 nM T00176 C2YPK9 44606647 Ki = 15.4 nM T00176 C5R8HZ 44608507 IC50 = 1800 nM T00176 C7OYC3 44825260 Ki = 916 nM T00176 CM8W5D 45138355 IC50 = 56 nM T00176 CQ0U7T 45139212 IC50 = 196 nM T00176 CA26FT 45139217 IC50 = 22 nM T00176 C3AX8L 45482969 IC50 = 140 nM T00176 CL68QB 46227513 IC50 > 100000 nM T00176 CZ2T0B 46840819 IC50 = 2.2 nM T00176 CL65SK 46840822 IC50 = 2.4 nM T00176 C2ZP7F 46894143 IC50 = 62500 nM T00176 CB62MX 49867311 Ki = 3 nM T00176 CE3P1T 50996417 IC50 = 8 nM T00176 CYG76I 51349561 IC50 = 69000 nM T00176 CB9GZ4 51349562 IC50 > 20000 nM T00176 CW2AC8 51349563 IC50 = 4200 nM T00176 CHC96B 51349698 IC50 = 4500 nM T00176 CYQ1E6 51349699 IC50 > 20000 nM T00176 CA45VB 51349700 IC50 = 15000 nM T00176 CWUJ19 51349701 IC50 = 6000 nM T00176 C25VAY 51349702 IC50 = 87000 nM T00176 C6JNQ7 51349703 IC50 = 9500 nM T00176 C2V6HS 51349704 IC50 = 2400 nM T00176 C63QZL 51349834 IC50 = 3100 nM T00176 C4SN3O 51349835 IC50 = 54000 nM T00176 C5ZUM9 51349836 IC50 = 7200 nM T00176 CK27ND 51349837 IC50 = 6200 nM T00176 CDM09A 51349838 IC50 = 6200 nM T00176 C6G3HF 51349839 IC50 = 47000 nM T00176 CYE21Q 51349840 IC50 > 100000 nM T00176 C3AO0Q 51349847 IC50 = 1300 nM T00176 C73PEB 51349971 IC50 > 20000 nM T00176 CTM3V8 51349972 IC50 > 100000 nM T00176 C7C2ET 51349973 IC50 > 100000 nM T00176 CCG4U1 51349974 IC50 > 100000 nM T00176 C2M1JN 51349975 IC50 > 100000 nM T00176 CSD95B 51349976 IC50 = 11000 nM T00176 CCBH37 51350114 IC50 > 100000 nM T00176 C1QM3O 51350115 IC50 = 88000 nM T00176 C9B3AE 51350116 IC50 > 20000 nM T00176 CZEQ91 51350117 IC50 > 20000 nM T00176 CKED96 51350118 IC50 > 200000 nM T00176 CIS2K0 51350119 IC50 > 200000 nM T00176 CW7ZS0 51350120 IC50 > 200000 nM T00176 CX2Z4O 51350252 IC50 > 200000 nM T00176 CV9P5I 51350253 IC50 > 200000 nM T00176 C39ORT 51350512 IC50 = 900 nM T00176 C8X0NF 51350513 IC50 = 1400 nM T00176 C0PUI1 51350514 IC50 = 570 nM T00176 C19MPN 51350515 IC50 = 980 nM T00176 CV2EA4 51350516 IC50 = 580 nM T00176 CCN9X6 51350650 IC50 = 730 nM T00176 CJ6B5D 51350651 IC50 = 570 nM T00176 CDBX96 51350652 IC50 = 390 nM T00176 C9PA3O 51350653 IC50 = 310 nM T00176 C9R0MG 51350782 IC50 = 1800 nM T00176 CB7D5O 51350783 IC50 = 2600 nM T00176 C4W1DG 51350784 IC50 = 2300 nM T00176 C7JM6L 51350785 IC50 = 1200 nM T00176 CI1T4X 51350786 IC50 = 1500 nM T00176 CB0ND4 51350787 IC50 = 2300 nM T00176 CMD09P 51350892 IC50 = 2800 nM T00176 CJLI15 51350893 IC50 = 8900 nM T00176 C6CP1E 51350894 IC50 = 8800 nM T00176 CCZ94I 51350895 IC50 = 49000 nM T00176 CY92NR 51350896 IC50 = 47000 nM T00176 CUR3J1 51351003 IC50 = 214000 nM T00176 C6GR4L 51351004 IC50 = 175000 nM T00176 C09XTY 51351005 IC50 > 20000 nM T00176 C72VHX 51351006 IC50 > 20000 nM T00176 CUK32E 51351007 IC50 > 50000 nM T00176 CZIY26 51351127 IC50 = 17000 nM T00176 C5RU9O 51351128 IC50 > 100000 nM T00176 CI0ZS8 51351129 IC50 = 252000 nM T00176 CZKP47 51351130 IC50 = 29000 nM T00176 C93VHI 51351131 IC50 = 11000 nM T00176 C6Y4AS 51351257 IC50 > 200000 nM T00176 C04IZE 51351258 IC50 > 200000 nM T00176 C0NT9M 51351259 IC50 = 33000 nM T00176 CXE65U 52943865 IC50 = 209000 nM T00176 CIUC38 53238217 IC50 = 5 nM T00176 C59UNR 53317544 IC50 = 6.2 nM T00176 CC15QU 53317691 IC50 = 170 nM T00176 CWCR13 53318463 IC50 > 20000 nM T00176 CNS1M9 53318519 IC50 = 400 nM T00176 CNX8V1 53318520 IC50 = 230 nM T00176 C86FIR 53318521 IC50 > 50000 nM T00176 C1Q8TB 53318829 IC50 = 28 nM T00176 CI08RL 53321450 IC50 = 77 nM T00176 C3ML7J 53321451 IC50 < 31 nM T00176 CR90KG 53321452 IC50 < 48 nM T00176 C1PUJ8 53322462 Ki = 170 nM T00176 CCV52T 53322772 IC50 < 10 nM T00176 C78AKT 53322773 IC50 = 1600 nM T00176 CTFZ46 53322774 IC50 < 48 nM T00176 CQEB58 53322938 IC50 = 2300 nM T00176 CBS75X 53323820 IC50 > 20000 nM T00176 CI9H2K 53325414 IC50 = 44 nM T00176 CMT70F 53325415 IC50 = 61 nM T00176 CZL74M 53358566 IC50 = 23 nM T00176 CM0Q2T 53358687 IC50 = 21 nM T00176 CY0MF5 53358688 IC50 = 25 nM T00176 CYE0S8 53470410 Ki = 250 nM T00176 C13JIF 53477213 Ki = 0.44 nM T00176 CKN24Z 56591348 IC50 = 1100 nM T00176 CQ8Y7H 56591370 IC50 = 18100 nM T00176 CJ9YQ2 56649312 IC50 = 7 nM T00176 CZW8C2 56839179 Ki = 130 nM T00176 CTN75O 56840663 Ki = 6700 nM T00176 C7NOC8 56846713 Ki = 400 nM T00176 C1V7OA 56941076 IC50 = 25 nM T00176 CV6Y9U 56941231 IC50 = 45 nM T00176 CF2O4I 56941233 IC50 = 7 nM T00176 CDGZ07 56941521 IC50 = 52 nM T00176 CI0T9D 56941522 IC50 = 140 nM T00176 CZ7RX8 56941669 IC50 = 52 nM T00176 C5Z4WC 56941811 IC50 = 11 nM T00176 CQXL07 56941947 IC50 = 47 nM T00176 C49PIE 56941948 IC50 = 6 nM T00176 CJ0HX2 56942230 IC50 = 18 nM T00176 C1SWU7 56942232 IC50 = 46 nM T00176 C4FV9E 56942233 IC50 = 52 nM T00176 C7KOV9 56942527 IC50 = 5764 nM T00176 C15HTM 56965957 IC50 = 1.1 nM T00176 CS9BE8 58006900 IC50 = 140 nM T00176 CX4F2J 58007119 IC50 = 11900 nM T00176 CF9R5T 58007373 IC50 = 15 nM T00176 COCH92 58007477 IC50 = 260 nM T00176 CV6X8S 58542331 IC50 = 1.2 nM T00176 C8KRY5 58573149 IC50 = 0.3 nM T00176 CNP0Q2 58573173 IC50 = 1.4 nM T00176 CYGZ76 58573255 IC50 = 0.5 nM T00176 C89AFP 58573438 IC50 = 0.3 nM T00176 CZO14M 58573543 IC50 = 0.091 nM T00176 CB5WF0 58573595 IC50 = 0.3 nM T00176 CN53OV 58573621 IC50 = 0.2 nM T00176 C9DXI7 58573665 IC50 = 1.3 nM T00176 CA1P3J 58573737 IC50 = 1.2 nM T00176 CHYP09 58573850 IC50 = 1.1 nM T00176 C56VCZ 58573852 IC50 = 0.7 nM T00176 C4H5WG 58573858 IC50 = 0.1 nM T00176 CW2AX3 58573904 IC50 = 0.2 nM T00176 C04KML 58894294 IC50 = 232 nM T00176 CY21UR 59249253 IC50 = 42 nM T00176 CUHA86 59249270 IC50 = 20 nM T00176 C06OQL 59249286 IC50 = 74 nM T00176 C0CZ8T 59249677 IC50 = 22 nM T00176 CEL4G7 59595061 IC50 = 2163 nM T00176 C04MIW 59647989 IC50 = 224 nM T00176 C3QSR9 59648009 IC50 = 334 nM T00176 C4OY6B 59648036 IC50 = 2700 nM T00176 C93DSA 59648084 IC50 = 492 nM T00176 CIF5X7 60154111 IC50 = 2400 nM T00176 CH6J8T 60156286 IC50 = 400 nM T00176 C32YBI 60167943 IC50 = 2 nM T00176 CVZ9M5 66760186 IC50 = 40 nM T00176 C21QNC 66760762 IC50 = 57 nM T00176 CW8G7T 66764524 IC50 = 177 nM T00176 CY5W7H 66987552 Ki = 6 nM T00176 C41OGA 67031670 IC50 = 25 nM T00176 CNW5H1 67032018 IC50 = 18 nM T00176 CQ54EG 67032045 IC50 = 4 nM T00176 C7O4TA 67032499 IC50 = 3 nM T00176 CL17FI 67034825 IC50 = 2 nM T00176 C7PZ8M 67035746 IC50 = 7 nM T00176 CLMC29 67035866 IC50 = 11 nM T00176 C8O5RY 67058380 IC50 = 21 nM T00176 C7PCK0 67058381 IC50 = 7.6 nM T00176 CLS1A3 67954173 IC50 = 4 nM T00176 CO0D3M 67954174 IC50 = 3 nM T00176 CG4RF2 67954180 IC50 = 6 nM T00176 CD8BR7 67954414 IC50 = 120 nM T00176 CAF98C 67954546 IC50 = 6 nM T00176 C7TV3K 67998850 IC50 = 0.64 nM T00176 CO3D4G 67998895 IC50 = 0.7 nM T00176 C4L7WM 67998916 IC50 = 0.2 nM T00176 C29YUV 67998930 IC50 = 0.2 nM T00176 CHA0I1 67999393 IC50 = 0.9 nM T00176 CBC6X9 67999477 IC50 = 0.2 nM T00176 C4T3IV 67999497 IC50 = 0.2 nM T00176 C3FC0S 67999720 IC50 = 0.096 nM T00176 C2QVS6 67999750 IC50 = 1.4 nM T00176 C41FZP 67999919 IC50 = 0.1 nM T00176 CGNB85 68000050 IC50 = 0.98 nM T00176 CI3YS0 68000097 IC50 = 0.098 nM T00176 CV53YR 68000111 IC50 = 0.3 nM T00176 CMK29V 68000113 IC50 = 0.2 nM T00176 C04ICY 68000346 IC50 = 62.4 nM T00176 CQU1F5 68000585 IC50 = 0.2 nM T00176 CW7Y0S 68000593 IC50 = 0.1 nM T00176 C3F9SN 68000685 IC50 = 0.2 nM T00176 CXWZ20 68000692 IC50 = 0.1 nM T00176 C4YO0Z 68000797 IC50 = 0.6 nM T00176 CVQ86U 68000913 IC50 = 0.4 nM T00176 C1X3ZP 68001022 IC50 = 0.3 nM T00176 C4HEC3 68001087 IC50 = 0.1 nM T00176 CCMG07 68805209 IC50 = 3000 nM T00176 CD4N0K 68806861 IC50 = 1100 nM T00176 C8MQP6 68807602 IC50 = 9500 nM T00176 CUQ2F5 68954893 IC50 = 7100 nM T00176 CUK0Q2 69498017 Ki = 0.86 nM T00176 CV7TU2 69498032 IC50 = 9.4 nM T00176 C8PT9A 70677271 Ki = 0.16 nM T00176 CL5XJ3 70682866 Ki = 8180 nM T00176 CNC09E 70682867 Ki = 89 nM T00176 CHXW50 70682883 Ki = 11900 nM T00176 CB24OY 70682884 Ki > 100000 nM T00176 CUTJ52 70684931 Ki > 100000 nM T00176 CH7WE9 70687100 Ki = 91 nM T00176 C4WI6K 70689172 Ki = 707 nM T00176 CWSU49 70689181 Ki = 315 nM T00176 C26VQK 70689182 Ki > 100000 nM T00176 CLHI31 70689192 Ki = 21100 nM T00176 CENC76 70693374 Ki = 721 nM T00176 CO4U0H 70693378 Ki = 3020 nM T00176 CRU40M 70693379 Ki = 1050 nM T00176 CF7HB8 70695473 Ki = 1370 nM T00176 CE04KX 70695481 Ki = 1720 nM T00176 CLS0P2 70695482 Ki > 100000 nM T00176 C6X2LU 70697491 Ki > 100000 nM T00176 CB6E2U 70697500 Ki = 37700 nM T00176 CXZ2M8 70697501 Ki = 3980 nM T00176 C02ROC 70697502 Ki = 518 nM T00176 CFB5H4 70872023 Ki = 2.9 nM T00176 CTO94S 70872137 Ki < 1 nM T00176 CQ63YN 71020635 Ki = 4.3 nM T00176 CNSA01 71020638 Ki = 1.7 nM T00176 C5QE1S 71020640 Ki = 1 nM T00176 CG70SP 71020641 Ki < 1 nM T00176 C97SJY 71020642 Ki < 1 nM T00176 CWJ4K3 71020643 Ki = 77 nM T00176 C04EPG 71020645 Ki = 1.2 nM T00176 CV17CM 71020646 Ki = 2.5 nM T00176 CW93BF 71020647 Ki = 3.4 nM T00176 CP5TO0 71020649 Ki = 3.4 nM T00176 CB2W1V 71020651 Ki = 12.8 nM T00176 C91FXI 71020652 Ki < 1 nM T00176 C6RJ8G 71020663 Ki = 4.5 nM T00176 C5TLD7 71020666 Ki < 1 nM T00176 C32EFX 71020667 Ki = 2.2 nM T00176 C5CYL2 71020668 Ki < 1 nM T00176 CL0KQ5 71020670 Ki < 1 nM T00176 CM2Y9T 71023078 IC50 > 2000 nM T00176 C62TRQ 71023080 Ki = 525 nM T00176 CSHU91 71023081 Ki < 1 nM T00176 C8GTF7 71023085 Ki = 19 nM T00176 CE8V3K 71023095 Ki = 2.8 nM T00176 CT28XM 71023130 Ki = 75.9 nM T00176 CB70QJ 71023133 IC50 > 2000 nM T00176 CQ46AN 71023161 Ki = 3.7 nM T00176 CAGM89 71023162 Ki = 9.8 nM T00176 C2AQT6 71023165 Ki = 1.7 nM T00176 C90DMG 71023185 Ki = 22 nM T00176 C6VU4Z 71023192 Ki = 15 nM T00176 CI6GS5 71305070 IC50 = 1000 nM T00176 CQ6CJ1 71305071 IC50 = 1800 nM T00176 COGY08 71305072 IC50 = 86 nM T00176 CISW47 71305074 IC50 = 610 nM T00176 CO9M5K 71449443 IC50 = 4400 nM T00176 CJ34RS 71451237 IC50 = 140 nM T00176 C2Z0OJ 71453053 IC50 = 1800 nM T00176 CR5E8Q 71453054 IC50 = 1200 nM T00176 CC1VW5 71453812 Ki = 260 nM T00176 CHQT69 71456576 IC50 = 2700 nM T00176 C6Q9NK 71458425 IC50 = 3100 nM T00176 CGZ6S2 71458426 IC50 = 840 nM T00176 C0YCM3 71544022 IC50 = 140 nM T00176 C60FEX 71544420 IC50 = 160 nM T00176 CC9H1S 71585475 IC50 = 7800 nM T00176 C6U8LX 71655426 IC50 = 52 nM T00176 CBJQ59 71663150 IC50 = 5400 nM T00176 CRA95Z 71663151 IC50 > 30000 nM T00176 C5MES9 71663332 IC50 > 30000 nM T00176 C1XD6G 71663333 IC50 = 1500 nM T00176 C6E0GY 71663334 IC50 = 1800 nM T00176 C0I5LP 71663335 IC50 = 1900 nM T00176 CUP8O4 71663336 IC50 = 2100 nM T00176 CTO9Y6 71663525 IC50 = 11700 nM T00176 CSW4E6 71663526 IC50 = 1800 nM T00176 CV02YU 71663527 IC50 > 30000 nM T00176 C7WV0H 71663528 IC50 = 1400 nM T00176 C7QOX3 71663529 IC50 = 880 nM T00176 CBLH41 71663696 IC50 = 100 nM T00176 CU8KD5 71663697 IC50 = 9900 nM T00176 CGV21W 71663698 IC50 = 1300 nM T00176 C4VZ2Y 71663699 IC50 = 7400 nM T00176 C12OST 71663864 IC50 = 16700 nM T00176 CCK36W 71678601 IC50 = 0.22 nM T00176 CI4ZS6 71678942 IC50 = 9500 nM T00176 C5E6HW 71678945 IC50 = 0.08 nM T00176 CA6Y9N 71716517 IC50 = 27500 nM T00176 C3D6JQ 71717127 IC50 = 8100 nM T00176 CKY7V2 71717128 IC50 = 14100 nM T00176 CP7C6V 71717752 IC50 > 30000 nM T00176 COJN30 71720163 IC50 > 30000 nM T00176 CA8F3J 71722565 Ki = 2000 nM T00176 CX35WQ 71722566 Ki = 43000 nM T00176 CKX5H9 71722568 Ki = 33000 nM T00176 C3FON5 71722717 Ki = 35000 nM T00176 CI6U2Y 71722718 Ki = 54000 nM T00176 CI5S4Q 71723197 Ki = 60000 nM T00176 CQ24PK 71745133 Ki = 0.62 nM T00176 C1A5HC 71747669 Ki = 0.61 nM T00176 CT07ZS 71747852 Ki = 0.94 nM T00176 CR09TV 71747853 Ki = 0.62 nM T00176 C5N9HJ 71747854 Ki = 2.4 nM T00176 CW3JG1 71777715 Ki = 1200 nM T00176 C7TIJ1 71818716 IC50 > 100000 nM T00176 CE4S1N 72697714 IC50 > 100000 nM T00176 CZI1E8 72697715 IC50 > 50000 nM T00176 CSJT35 72697716 IC50 > 100000 nM T00176 CL2P0H 72697717 IC50 > 100000 nM T00176 CE94TV 72697718 IC50 > 100000 nM T00176 CG8K9U 72697719 IC50 > 100000 nM T00176 CTR16S 72697857 IC50 > 100000 nM T00176 C9IJH3 72697858 IC50 > 100000 nM T00176 CK3DA4 72697859 IC50 > 100000 nM T00176 CKC91P 72714997 IC50 = 22200 nM T00176 CN75KD 72714998 IC50 = 21300 nM T00176 CPK9C0 73297272 IC50 = 5.57 nM T00176 CH15WP 73345928 Ki = 250 nM T00176 CG5X1Q 73347121 IC50 = 3000 nM T00176 CY9UN4 73347446 Ki = 80 nM T00176 C3W1YC 73347473 IC50 = 214 nM T00176 CME7R0 73348988 IC50 = 8510 nM T00176 CZ5SJ0 73349557 IC50 = 1500 nM T00176 C28XBR 73349627 IC50 = 49500 nM T00176 CC1HZ5 73349628 IC50 = 12300 nM T00176 CHUA84 73351169 IC50 > 100000 nM T00176 CHUZ81 73354083 IC50 = 10700 nM T00176 C9BEI4 73354084 IC50 = 11900 nM T00176 CFJ72A 73355609 IC50 = 17500 nM T00176 C7RT2B 73355682 IC50 > 100000 nM T00176 CU47MB 73355683 IC50 = 15000 nM T00176 CVFR62 73356477 IC50 = 8900 nM T00176 CPQ3H1 73357201 IC50 = 32000 nM T00176 CE5PO4 73357202 IC50 = 8400 nM T00176 CRE7I6 73386674 IC50 = 2 nM T00176 C7XN3A 73386675 IC50 = 0.1 nM T00176 CZQV24 73386676 IC50 = 0.1 nM T00176 CT64FE 73386677 IC50 = 0.1 nM T00176 C1TY5X 73386678 IC50 = 0.1 nM T00176 CFZ7E0 73386679 IC50 = 9 nM T00176 C8UB4G 76310907 IC50 = 0.5 nM T00176 CAJ9E5 76318138 IC50 = 0.7 nM T00176 C5DY6V 76321813 IC50 = 0.1 nM T00176 C5A9VY 76321823 IC50 = 5.6 nM T00176 CZCW30 76325459 IC50 = 1.2 nM T00176 C3P2OS 76328371 IC50 = 33 nM T00176 C40PHT 76328991 IC50 = 1.3 nM T00176 CU81GN 76328992 IC50 = 0.1 nM T00176 CQ8UW4 76329003 IC50 = 0.1 nM T00176 CF4YD7 76329004 IC50 = 0.9 nM T00176 C34NUV 76332045 IC50 = 17 nM T00176 CHB16Z 76332677 IC50 = 0.1 nM T00176 C3CHB8 76336278 IC50 = 0.2 nM T00176 C7DPL0 77108133 IC50 = 0.6 nM T00176 C0B3ZQ 77461139 IC50 = 1000 nM T00176 CN52SO 78147351 IC50 = 0.16 nM T00176 CR2TL5 85468775 Ki > 25000 nM T00176 CNRQ94 86298586 Ki = 90 nM T00176 C2V8YN 86298587 Ki = 90 nM T00176 CP7YN8 86730799 IC50 = 0.9 nM T00176 CE3U4D 86730805 IC50 = 1.1 nM T00176 C7XU0W 86731821 IC50 = 0.37 nM T00176 CZSU26 86731830 IC50 = 0.1 nM T00176 CNB31V 86766851 IC50 = 0.14 nM T00176 CRCZ56 86766852 IC50 = 0.17 nM T00176 CJCY10 86766868 IC50 = 0.26 nM T00176 CB13DK 86766904 IC50 = 13 nM T00176 C0F6IP 87252745 IC50 = 15 nM T00176 CTHD96 87252803 IC50 = 11 nM T00176 C9NA4J 89478355 IC50 = 0.8 nM T00176 CKT75Q 89478490 IC50 = 0.4 nM T00176 C73NTD 89478498 IC50 = 1.3 nM T00176 CR8G1A 89478524 IC50 = 3 nM T00176 C8Y3MJ 89478729 IC50 = 17 nM T00176 C3S4EZ 89480425 IC50 = 2 nM T00176 C32RUJ 89480496 IC50 = 0.5 nM T00176 C1UA5H 89490679 IC50 = 1.1 nM T00176 C2USI5 89490693 IC50 = 5 nM T00176 CHB05N 89490787 IC50 = 20 nM T00176 C8R4OB 89490809 IC50 = 18 nM T00176 C62GRI 89490890 IC50 = 2 nM T00176 CM9X5R 89601404 IC50 = 0.13 nM T00176 C3W7PA 90342080 IC50 = 2.3 nM T00176 CV0XI5 90342165 IC50 = 0.5 nM T00176 CE91KJ 90342208 IC50 = 0.6 nM T00176 CN95OP 90347747 IC50 = 0.4 nM T00176 CS2IZ9 90347748 IC50 = 0.3 nM T00176 CE2XU8 90354304 IC50 = 0.1 nM T00176 CI0AL1 90368833 IC50 = 0.13 nM T00176 CH0PN3 90643708 Ki = 340 nM T00176 C5WR7Q 90643709 Ki = 280 nM T00176 CBXT49 90643710 Ki = 240 nM T00176 C86YXR 90643711 Ki = 200 nM T00176 CGO12D 90643712 Ki = 150 nM T00176 C3X8HK 90643713 Ki = 140 nM T00176 CD8M0A 90643714 Ki = 190 nM T00176 C1KP0N 90643715 Ki = 140 nM T00176 C8D5RE 90643716 Ki = 100 nM T00176 C1RP4V 90643717 Ki = 230 nM T00176 CV2BG6 90644126 Ki = 1370 nM T00176 CZK05E 90644127 Ki > 100000 nM T00176 CL85PM 90644128 Ki = 720 nM T00176 CY6UF5 90644129 Ki = 710 nM T00176 CYC9W3 90644130 Ki > 100000 nM T00176 C36HUT 90644131 Ki = 1720 nM T00176 C8SHC6 90644132 Ki = 320 nM T00176 COT89H 90644133 Ki = 8180 nM T00176 CQY63Z 90644134 Ki = 3020 nM T00176 C7W9RZ 90644135 Ki > 100000 nM T00176 CRG49C 90644136 Ki > 100000 nM T00176 C5VAN2 90644137 Ki = 37700 nM T00176 CB1N9A 90644138 Ki = 150 nM T00176 C2VDW8 90644646 IC50 = 24 nM T00176 C1S8PM 90644647 IC50 = 24 nM T00176 C5WDB0 90644648 IC50 = 24 nM T00176 C65BZC 90644878 IC50 = 360 nM T00176 CSX7N6 90644879 IC50 = 440 nM T00176 C8NF1O 90644880 IC50 = 810 nM T00176 CWAT67 90644881 IC50 = 780 nM T00176 CV5G6C 90644882 IC50 = 610 nM T00176 C0YG7F 90644883 IC50 = 570 nM T00176 C1AHE4 90644884 IC50 = 550 nM T00176 CY2QZ0 90644885 IC50 = 260 nM T00176 C6R4QV 90654509 IC50 = 600 nM T00176 CF72HM 90654510 IC50 = 300 nM T00176 CK5NW8 90654511 IC50 = 4000 nM T00176 C5DPB9 90654512 IC50 = 3000 nM T00176 CB54FD 90654513 IC50 = 3900 nM T00176 CPAD85 90654514 IC50 > 10000 nM T00176 CP8JX2 90654515 IC50 = 5600 nM T00176 CV09GW 90655372 IC50 = 0.1 nM T00176 CB2RM8 90655373 IC50 = 0.2 nM T00176 CHBG56 90655374 IC50 = 0.8 nM T00176 C0NXS3 90655376 IC50 = 3.1 nM T00176 CV72RT 90655377 IC50 = 1.9 nM T00176 CF68GW 90655378 IC50 = 3.7 nM T00176 CNBZ28 90655379 IC50 = 0.5 nM T00176 C26LUH 90655380 IC50 = 1.1 nM T00176 CZD14Q 90655381 IC50 = 1.8 nM T00176 C4OCF1 90655382 IC50 = 0.1 nM T00176 COBZ93 90655383 IC50 = 0.3 nM T00176 CT4ZL3 90655384 IC50 = 7.6 nM T00176 COZS39 90655385 IC50 = 0.1 nM T00176 C5HKB1 90655386 IC50 = 1.2 nM T00176 CD3R7I 90655387 IC50 = 0.1 nM T00176 C3X7VT 90655388 IC50 = 0.2 nM T00176 CU76JS 90655389 IC50 = 1.7 nM T00176 C6U5AF 90655390 IC50 = 0.4 nM T00176 C0PL1S 90655391 IC50 = 5.9 nM T00176 C20JNZ 90655392 IC50 = 0.1 nM T00176 CGV6B3 90655393 IC50 = 0.1 nM T00176 CUK5G7 90655394 IC50 = 0.1 nM T00176 C4RMZ5 90655395 IC50 = 3 nM T00176 CQK5U3 90655396 IC50 = 0.1 nM T00176 CZB2Q5 90655397 IC50 = 8.1 nM T00176 CO5H9B 90655398 IC50 = 0.1 nM T00176 CB68UJ 90655399 IC50 = 0.1 nM T00176 CH9EN4 90655400 IC50 = 0.3 nM T00176 CX5TE2 90655401 IC50 = 0.1 nM T00176 C17PXB 90655402 IC50 = 2.1 nM T00176 CCA0O4 90655403 IC50 = 0.2 nM T00176 C8Y5CE 90655404 IC50 = 0.1 nM T00176 CQC65V 90655405 IC50 = 0.1 nM T00176 CG2S6U 90655406 IC50 = 0.1 nM T00176 C9G0KC 90655407 IC50 = 0.1 nM T00176 C68YUI 90655408 IC50 = 0.2 nM T00176 C3W9PH 90655409 IC50 = 8 nM T00176 CHUS42 90656493 Ki = 1800 nM T00176 CWT8K7 90656494 Ki = 600 nM T00176 C6D7NR 90666823 IC50 = 700 nM T00176 CKA25D 90666824 IC50 = 1900 nM T00176 C45OVU 90666825 IC50 = 1900 nM T00176 CKGW70 90666826 IC50 = 4700 nM T00176 CE89VR 90666827 IC50 = 200 nM T00176 CS93YN 90666828 IC50 = 300 nM T00176 CAP95E 90666829 IC50 = 890 nM T00176 C98YWK 90666830 IC50 = 260 nM T00176 CIT5X4 90666831 IC50 = 17000 nM T00176 C8RI2H 90666832 IC50 = 2900 nM T00176 C7FKE1 90666833 IC50 > 50000 nM T00176 C3Z8WE 90666834 IC50 = 2900 nM T00176 C03GLI 90666835 IC50 = 2500 nM T00176 CE5FT8 90666836 IC50 = 7600 nM T00176 CL9H7W 90666837 IC50 = 15000 nM T00176 CP5GD7 90666838 IC50 = 17000 nM T00176 CLA53P 90666839 IC50 = 760 nM T00176 CU91QC 90666840 IC50 = 1100 nM T00176 C5W9VY 90666841 IC50 = 1600 nM T00176 CPJ8A5 90666842 IC50 = 1600 nM T00176 CLV12D 90667000 IC50 = 2100 nM T00176 C82EPU 90667001 IC50 = 2200 nM T00176 C0FG5C 90667002 IC50 = 190 nM T00176 CXEK45 90681222 IC50 = 169 nM T00176 C8H4KE 90681223 IC50 = 41 nM T00176 C0XL7P 91668261 IC50 = 0.22 nM T00176 C5T9WD 94962278 Ki = 2290 nM T00176 CJD64H 117884868 Ki = 3.4 nM T00176 CU84PT 117884873 Ki = 19 nM T00176 CS15TR 118458373 Ki < 1 nM T00176 C9OP6I 118458374 Ki < 1 nM T00176 CVA2Y4 118458376 Ki = 1.3 nM T00176 CBL35M 118458378 Ki < 1 nM T00176 CL78ZQ 118459062 Ki < 1 nM T00176 CP4W2R 118709118 IC50 = 0.079 nM T00176 CBC17J 118709119 IC50 = 0.11 nM T00176 C1ZU4M 118709120 IC50 = 0.081 nM T00176 CN3Y9V 118709121 IC50 = 0.17 nM T00176 C6I4CK 118709122 IC50 = 0.059 nM T00176 CQ5W4O 118709123 IC50 = 0.086 nM T00176 CSG60B 118709124 IC50 = 0.12 nM T00176 C91VXE 118709125 IC50 = 0.15 nM T00176 C3WEV7 118709126 IC50 = 0.071 nM T00176 C2C6OE 118709127 IC50 = 0.12 nM T00176 C7TBO9 118709128 IC50 = 0.16 nM T00176 C5RU6X 118709129 IC50 = 0.075 nM T00176 C26FCE 118709130 IC50 = 0.53 nM T00176 C7U1YJ 118709131 IC50 = 0.3 nM T00176 CJ43KH 118709132 IC50 = 0.31 nM T00176 C2KCO5 118709133 IC50 = 0.24 nM T00176 C4RHD3 118709134 IC50 = 0.4 nM T00176 C0VN5J 118709135 IC50 = 0.38 nM T00176 CLDU10 118709136 IC50 = 0.47 nM T00176 C4P8QS 118709137 IC50 = 0.15 nM T00176 CW1Q4Z 118709138 IC50 = 1.1 nM T00176 CUMF74 118709139 IC50 = 0.074 nM T00176 CP30UF 118709140 IC50 = 0.088 nM T00176 C8FE4G 118709141 IC50 = 0.059 nM T00176 C74UXE 118709142 IC50 = 0.37 nM T00176 CS0J5F 118709143 IC50 = 0.42 nM T00176 CFI1P5 118709144 IC50 = 0.12 nM T00176 CC3FL7 118718047 IC50 = 150 nM T00176 CNQT35 118718079 Ki = 5 nM T00176 CPC03Z 118720811 Ki = 105 nM T00176 CV29CT 118720812 Ki = 234 nM T00176 CCR61H 118720813 Ki = 1301 nM T00176 C5GSE8 118720814 Ki = 80 nM T00176 CRX7A9 118720815 Ki = 23 nM T00176 CG2JC8 118720816 Ki = 1238 nM T00176 CEI1K0 118720817 Ki = 67 nM T00176 CR8V2D 118720818 Ki = 3 nM T00176 CTP36N 118720819 Ki = 1026 nM T00176 C81ORY 118720820 Ki = 53 nM T00176 CJ30PY 118720821 IC50 > 10000 nM T00176 CNW2V3 118730174 IC50 < 0.1 nM T00176 CL46FO 118730175 IC50 = 0.18 nM T00176 C4YAB3 118730176 IC50 = 0.18 nM T00176 CT96NZ 118730177 IC50 = 0.21 nM T00176 CNZC46 118730178 IC50 = 0.37 nM T00176 C1RYW3 118730179 IC50 = 0.49 nM T00176 CLD90T 118730180 IC50 = 2.4 nM T00176 CCL9V8 118730181 IC50 = 0.21 nM T00176 CKGR58 118730182 IC50 = 0.21 nM T00176 C05DSN 118730183 IC50 = 1.8 nM T00176 C3B6MC 118730184 IC50 = 0.42 nM T00176 C16YJR 118730185 IC50 < 0.1 nM T00176 CUK7G6 118730186 IC50 = 0.79 nM T00176 CO30CN 118730187 IC50 = 0.49 nM T00176 CB57YK 118730188 IC50 = 0.52 nM T00176 C90KHE 118730189 IC50 = 0.26 nM T00176 CE9D2H 118730190 IC50 = 0.5 nM T00176 C2DGC3 122192870 Ki = 3050 nM T00176 CB73VQ 122192871 Ki = 6960 nM T00176 C8C0XM 122192873 Ki = 690 nM T00176 C2ZT4V 122192874 Ki = 360 nM T00176 C3RON1 122192875 Ki = 710 nM T00176 CS8XT3 122192876 Ki = 7220 nM T00176 C3W8YL 122192877 Ki = 1820 nM T00176 CFHE72 122689625 IC50 = 43 nM T00176 C95MAK 126963310 Ki = 58 nM T00176 C6I9MQ 127035023 Ki = 17000 nM T00176 CSI49A 127035024 Ki = 10000 nM T00176 CD0Q5H 127035025 Ki > 22000 nM T00176 CFZ35L 127035026 Ki = 6700 nM T00176 CFK31G 127035027 Ki = 1800 nM T00176 CVY7S6 127035701 Ki = 700 nM T00176 CF86ES 127035702 Ki > 60000 nM T00176 C0N9ES 127045680 IC50 = 267 nM T00176 C9MWP5 127045711 IC50 = 801 nM T00176 C80FRK 127045712 IC50 = 4026 nM T00176 C63PWT 127045713 Ki = 1130 nM T00176 CU75LD 127045714 Ki = 689 nM T00176 CV4K2N 127045715 Ki = 301 nM T00176 C9TS4I 127045716 Ki = 446 nM T00176 C2PNY9 127045860 IC50 = 399 nM T00176 CM2R5I 127045886 IC50 = 1065 nM T00176 CZ2GC1 127045923 IC50 = 7744 nM T00176 C8AU5I 127045924 IC50 = 111 nM T00176 CUT8S3 127045927 Ki = 107 nM T00176 CS5N1J 127046058 IC50 = 2400 nM T00176 C3SZ6J 127046167 IC50 = 144 nM T00176 C5F1VM 127046265 IC50 = 1981 nM T00176 C9TEH7 127046266 IC50 = 8766 nM T00176 CAS76F 127046360 IC50 = 8721 nM T00176 C1LO3T 127046361 IC50 = 4276 nM T00176 CT90WN 127046362 IC50 = 114 nM T00176 C83QXA 127046501 IC50 = 293 nM T00176 C9IFO6 127046502 IC50 = 2399 nM T00176 CM06ON 127046503 IC50 = 173 nM T00176 CVEJ14 127046716 Ki = 422 nM T00176 CZWO41 127046726 IC50 = 392 nM T00176 C57ZRE 127046727 IC50 = 42 nM T00176 C5LWC3 127046831 IC50 = 1919 nM T00176 CU7J1K 127046832 IC50 = 150 nM T00176 C4F2JM 127046867 Ki = 4470 nM T00176 C8R2OD 127046868 Ki = 2190 nM T00176 CW7KI2 127046869 Ki = 4280 nM T00176 C93DAC 127046910 IC50 = 5831 nM T00176 CPB9D6 127046994 IC50 = 2039 nM T00176 C5LX0Y 127046995 IC50 = 2359 nM T00176 CZO61I 127046996 IC50 = 1863 nM T00176 CA5VP1 127046997 IC50 = 686 nM T00176 CZ8C3V 127047003 Ki = 7420 nM T00176 C4D6XB 127047004 Ki = 19800 nM T00176 CL68JY 127047005 Ki = 1030 nM T00176 CX6WE4 127047006 Ki = 712 nM T00176 C9FMI6 127047007 Ki = 2140 nM T00176 C9TCV7 127047008 Ki = 616 nM T00176 CISJ19 127047103 IC50 = 2764 nM T00176 CN68EI 127047104 IC50 = 2095 nM T00176 C0JN8G 127047105 IC50 = 4112 nM T00176 CQC09U 127047106 IC50 = 8714 nM T00176 CAV7T9 127047554 IC50 = 376 nM T00176 CW6XP0 127047555 IC50 = 525 nM T00176 CY9KS2 127047694 IC50 = 5027 nM T00176 CDPX03 127047695 IC50 = 1146 nM T00176 C27JEI 127047769 IC50 = 9359 nM T00176 CTZ34F 127047770 IC50 = 25801 nM T00176 CI69NG 127047771 IC50 = 6599 nM T00176 CJZ5G4 127047772 IC50 = 668 nM T00176 C4INZ2 127050965 IC50 = 154.6 nM T00176 C8MG9S 127050966 IC50 = 24.8 nM T00176 C34MQG 127050967 IC50 = 4.3 nM T00176 C8FHY7 127050968 IC50 = 9.8 nM T00176 C3F0BZ 127051540 IC50 = 11.65 nM T00176 C7YJG6 127051541 IC50 = 15.2 nM T00176 CR9OY5 127051542 IC50 = 77.7 nM T00176 CWL02R 127051543 IC50 = 11.7 nM T00176 C01WVT 136044100 IC50 = 890 nM T00176 C5YNB3 136044101 IC50 = 910 nM T00176 CC2F1W 136044102 IC50 = 940 nM T00176 C80WCI 136044103 IC50 = 970 nM T00176 C83QVU 136056460 IC50 = 1.3 nM T00176 C68JWY 136209736 IC50 = 17 nM T00176 CS28FE 136607458 IC50 = 990 nM T00176 CLQT37 136607459 IC50 = 840 nM T00176 C73CEN 137243602 Ki = 24300 nM T00176 CUOK03 137350181 Ki = 600 nM T00176 C3ZGV0 137631366 Ki = 157 nM T00176 C64ORN 137631715 Ki < 1 nM T00176 C6T1ZE 137632191 Ki = 1060 nM T00176 CJ6D2B 137632638 Ki = 3.1 nM T00176 CC3HQ7 137633155 IC50 = 93.7 nM T00176 CWY4X0 137633285 IC50 = 141.5 nM T00176 CGHT40 137633360 Ki = 26080 nM T00176 CR1LJ0 137634060 Ki = 20 nM T00176 C3KUO4 137634336 Ki = 6020 nM T00176 C5Q2IU 137634453 Ki = 2310 nM T00176 CF47DC 137634792 Ki = 650 nM T00176 C7GNM5 137634976 Ki = 2470 nM T00176 CF8O9P 137635775 Ki = 1 nM T00176 CTB94X 137635847 Ki = 130 nM T00176 CY6B5Q 137636017 Ki = 59 nM T00176 CQKB65 137636927 Ki = 63 nM T00176 CX83PQ 137637822 Ki = 1530 nM T00176 CZ31RB 137637908 IC50 = 9.2 nM T00176 C5JAR3 137637954 Ki = 1 nM T00176 C3V6SE 137638070 Ki = 30 nM T00176 CXC18M 137638774 Ki = 36570 nM T00176 CP1HD6 137639153 Ki = 23 nM T00176 C4ROS5 137639702 Ki = 60 nM T00176 CN8H7U 137639899 Ki = 13.7 nM T00176 C17SXB 137640724 IC50 = 50.3 nM T00176 CZBT67 137641354 Ki = 680 nM T00176 CD65PZ 137641635 Ki = 990 nM T00176 C0VID4 137642157 Ki = 1640 nM T00176 CN74GZ 137642196 Ki < 1 nM T00176 CQ8P1F 137642328 Ki = 60 nM T00176 CT9DS6 137642818 Ki = 860 nM T00176 CC13NQ 137644080 Ki = 170 nM T00176 CYJX38 137644563 Ki = 98 nM T00176 C1TYP0 137645068 Ki = 44000 nM T00176 C82UMH 137645566 Ki = 640 nM T00176 C0WHG9 137645614 Ki = 8 nM T00176 C6KQ3F 137645827 Ki = 520 nM T00176 CC7A2I 137646423 Ki = 15700 nM T00176 C0HE7C 137646573 Ki = 13.2 nM T00176 CH4IA7 137646610 Ki = 2.7 nM T00176 C61JDO 137646640 IC50 = 18.9 nM T00176 CLNB01 137646904 Ki = 121 nM T00176 CQLA87 137647053 Ki = 15 nM T00176 C43INM 137647313 IC50 = 23.4 nM T00176 CUL1O6 137647880 Ki = 50 nM T00176 CUJQ86 137648552 Ki = 170 nM T00176 CTG03A 137648583 Ki = 20 nM T00176 C6PZ7V 137648635 Ki < 1 nM T00176 CWB46V 137649150 Ki = 4890 nM T00176 CT52RE 137650048 Ki = 29 nM T00176 CE3V8Y 137650518 Ki = 17 nM T00176 C78BTI 137651111 Ki = 21 nM T00176 C5AR9B 137651117 Ki = 4380 nM T00176 COZN30 137651734 Ki = 120 nM T00176 C3KNQ1 137652580 Ki = 4.2 nM T00176 C97XEB 137652895 Ki = 970 nM T00176 CY4RZ6 137653137 IC50 = 52.4 nM T00176 C7KZ4L 137653948 IC50 = 115 nM T00176 CBW18Q 137653977 Ki = 6.5 nM T00176 CJAC03 137654113 Ki = 10870 nM T00176 C2OJU7 137654973 Ki = 656 nM T00176 CIC2K9 137655254 Ki = 433 nM T00176 CVP38H 137655392 Ki = 18140 nM T00176 C8R0UO 137655459 IC50 = 65.3 nM T00176 CP3FI9 137655549 Ki = 170 nM T00176 CWRU31 137655568 Ki = 38 nM T00176 C4HB1U 137656155 IC50 = 7.85 nM T00176 CUO17X 137656185 Ki = 1930 nM T00176 CR7WG9 137656205 Ki = 225 nM T00176 C2QHP5 137656534 IC50 = 35.4 nM T00176 CU3FN6 137657022 IC50 = 9.6 nM T00176 CBW6G3 137657187 Ki = 2.8 nM T00176 CPHT95 137657789 Ki = 322 nM T00176 CD1P0Y 137657895 Ki = 290 nM T00176 CN84DX 137658063 Ki = 230 nM T00176 C7QF5S 137658136 Ki = 54 nM T00176 CF41UL 137658356 Ki = 13.9 nM T00176 CJD09N 137658607 Ki = 2.4 nM T00176 CTM69S 137658613 Ki = 117000 nM T00176 CV14BP 137658881 Ki = 100 nM T00176 C49VQU 137658988 Ki = 200 nM T00176 CL32PN 137659377 Ki = 2.2 nM T00176 CDMY96 137659576 IC50 = 13.8 nM T00176 C17FTO 137659676 Ki = 90 nM T00176 CR6M4D 137660349 Ki = 1.9 nM T00176 CZ5T9H 137660352 Ki = 28000 nM T00176 C3JM5Y 137660704 Ki = 38 nM T00176 CP5Z3Q 137661363 Ki = 70 nM T00176 CF8IU3 137661501 Ki = 81.2 nM T00176 CHD18T 137661621 Ki = 21 nM T00176 CM7P2H 137661851 Ki = 80 nM T00176 CWJ84Q 137662288 Ki = 9520 nM T00176 C4NFS3 138393072 Ki = 110 nM T00176 C9XB0W 139600332 IC50 = 67.5 nM T00176 C1JMN9 145949196 Ki = 170 nM T00176 C3M7JG 145949513 Ki = 290 nM T00176 C0X8ER 145949722 IC50 = 270 nM T00176 CXEV29 145949841 Ki = 620 nM T00176 C1G2PB 145949937 Ki = 580 nM T00176 C39NQZ 145950005 Ki = 80 nM T00176 CF54HP 145950469 Ki = 1050 nM T00176 CI0MO1 145950501 Ki = 100 nM T00176 CMOW75 145951496 Ki = 960 nM T00176 C2MO7K 145951845 IC50 > 1000 nM T00176 CG80FB 145951878 IC50 = 624 nM T00176 CMZ58R 145952121 Ki = 1020 nM T00176 CT2W3K 145952145 Ki = 1800 nM T00176 C74YTI 145952178 Ki = 3000 nM T00176 CR57VX 145952811 Ki = 700 nM T00176 C1P0NL 145952828 IC50 = 72 nM T00176 CV5QI2 145952910 Ki = 330 nM T00176 CP13JE 145953191 Ki = 2500 nM T00176 CSY17G 145953588 Ki = 1900 nM T00176 CJA7N9 145953608 IC50 = 389 nM T00176 C39QEU 145954116 Ki = 5300 nM T00176 CZ4SK6 145954275 IC50 = 333 nM T00176 CYD83K 145954811 Ki = 10890 nM T00176 CJ7BQ3 145954848 Ki = 350 nM T00176 C4G8DC 145955221 Ki = 140 nM T00176 CUM12F 145956028 Ki = 57 nM T00176 CTA08K 145956036 IC50 = 370 nM T00176 CY5I1O 145956101 IC50 = 685 nM T00176 C8RAG3 145956154 IC50 = 308 nM T00176 CM6UC8 145956323 Ki = 280 nM T00176 CCB51L 145956802 IC50 = 720 nM T00176 CBED35 145957183 Ki = 70 nM T00176 CAP1Y3 145957299 Ki = 60 nM T00176 CS6K8G 145957478 Ki = 2650 nM T00176 C1R8DB 145957798 Ki = 170 nM T00176 CJZ25F 145958256 Ki = 260 nM T00176 CMY49F 145958259 Ki = 340 nM T00176 CTS5R3 145959048 IC50 = 437 nM T00176 C8RXN1 145959262 Ki = 1430 nM T00176 CTPK43 145959386 Ki = 320 nM T00176 CU78RJ 145959742 Ki = 460 nM T00176 CQ4ET5 145959752 IC50 > 1000 nM T00176 CH5VM4 145960138 Ki = 1300 nM T00176 CO0W4J 145961652 IC50 = 545 nM T00176 CP0U3W 145966080 Ki = 6700 nM T00176 CQRM37 145967267 Ki = 4000 nM T00176 CB17RI 145969823 Ki = 2600 nM T00176 C82QUX 145969865 Ki = 6100 nM T00176 C23HZY 145971531 IC50 > 1000 nM T00176 CFX6H0 145971585 Ki = 12000 nM T00176 CGOE24 145972301 Ki = 23000 nM T00176 CIU10W 145972713 Ki = 340 nM T00176 CY9M0G 145972753 Ki = 700 nM T00176 C2GM8B 145973174 Ki = 320 nM T00176 CRD8G6 145974350 Ki = 90 nM T00176 CIZ01H 145974418 Ki = 2800 nM T00176 C5IQ9T 145975898 Ki = 8200 nM T00176 C8WA9J 145976121 Ki = 7000 nM T00176 CUK8M4 145976465 Ki = 14000 nM T00176 C3SI0B 145976526 Ki = 9700 nM T00176 C4R2KX 145977314 Ki = 4400 nM T00176 C8LSJ7 145978249 Ki = 93000 nM T00176 C7DSC3 145980812 Ki = 400 nM T00176 CW7ZU8 145982231 Ki = 600 nM T00176 CX1MK3 145989243 IC50 = 0.26 nM T00176 CQ2F7W 145989532 IC50 = 0.074 nM T00176 CO41YV 145991230 Ki = 1200 nM T00176 CNH2T4 145992205 Ki = 200 nM T00176 CPF13W 145993071 Ki = 1900 nM T00176 C7C2PX 155511790 Ki = 1850 nM T00176 CJZ61W 155511975 IC50 = 4900 nM T00176 C8R7FV 155512750 IC50 = 1.2 nM T00176 C81LBF 155513253 Ki = 3440 nM T00176 C4L8IS 155514420 Ki = 0.88 nM T00176 CG5FX7 155515298 IC50 = 891 nM T00176 CFHN28 155516869 IC50 = 11.9 nM T00176 CWI45U 155517444 Ki = 720 nM T00176 C3PD6F 155518117 Ki = 11880 nM T00176 CX8S5M 155518427 IC50 > 20000 nM T00176 CH9CB8 155519596 IC50 = 600 nM T00176 CVS02D 155519704 IC50 = 4140 nM T00176 CNGH35 155521620 Ki = 1020 nM T00176 CZ21FA 155522131 Ki = 70 nM T00176 CCX4D5 155522186 Ki = 1630 nM T00176 CM5AP4 155522379 Ki = 11630 nM T00176 CZM5R1 155522380 Ki = 4000 nM T00176 C6YEG9 155523178 Ki = 4670 nM T00176 CB8G5R 155523298 Ki = 500 nM T00176 C78PNX 155523379 Ki = 34 nM T00176 C0HAV7 155524001 Ki = 320 nM T00176 CYM94J 155526750 Ki = 4802 nM T00176 C7N0SY 155526905 Ki = 740 nM T00176 CJC07B 155527872 IC50 = 3950 nM T00176 CI16PB 155528357 IC50 = 3220 nM T00176 C60AWK 155529405 Ki = 0.045 nM T00176 CWC32Z 155529926 Ki = 1680 nM T00176 C5R8YO 155530377 Ki = 300 nM T00176 CYL1M7 155532432 Ki = 2240 nM T00176 C2WB7O 155532959 Ki = 3280 nM T00176 CKUT47 155534630 Ki = 61 nM T00176 CQ65MS 155535133 IC50 = 10.5 nM T00176 CWGE76 155537056 IC50 = 3600 nM T00176 CJ9SV2 155539377 IC50 = 0.8 nM T00176 C9T2LU 155539551 Ki = 360 nM T00176 CZJ43Y 155540256 Ki = 620 nM T00176 C7AIS2 155540935 Ki = 2280 nM T00176 C5BLH7 155541232 IC50 = 1900 nM T00176 C4E6YV 155541314 Ki = 370 nM T00176 CS74BO 155541655 Ki = 390 nM T00176 C49XKD 155542750 Ki = 2300 nM T00176 C7DH4S 155542925 IC50 = 2800 nM T00176 CYXP56 155543879 IC50 = 10500 nM T00176 CR3SC8 155544506 Ki = 19800 nM T00176 CE20GK 155544614 IC50 > 20000 nM T00176 CUS85I 155546101 IC50 = 4610 nM T00176 CVG09H 155546326 Ki = 6 nM T00176 CD54OX 155546509 Ki = 240 nM T00176 C6R0OI 155546787 IC50 = 11.9 nM T00176 CV76YM 155547556 Ki = 260 nM T00176 CW8J1M 155548484 Ki = 420 nM T00176 CZTG39 155548608 Ki = 0.44 nM T00176 CH9K2S 155549013 IC50 > 20000 nM T00176 C7E9DQ 155550524 Ki = 420 nM T00176 C2BG3P 155553262 IC50 > 20000 nM T00176 CN34RO 155553441 IC50 = 1.2 nM T00176 CC5LD1 155554511 Ki = 570 nM T00176 CKOD46 155554714 Ki = 5280 nM T00176 CMI3L2 155555639 Ki = 6 nM T00176 C7ZF4U 155558272 Ki = 140 nM T00176 C7YWV8 155558664 Ki = 760 nM T00176 C0PR4Z 155558699 Ki = 34 nM T00176 CH72VR 155558976 Ki = 43800 nM T00176 C3DBH9 155559256 IC50 = 11.9 nM T00176 CH5N3K 155559422 Ki = 1720 nM T00176 CU8G5C 155559974 Ki = 3680 nM T00176 CSER69 155561097 Ki = 2540 nM T00176 C39FDU 155561757 IC50 = 24 nM T00176 C8J2DG 155562316 IC50 = 1400 nM T00176 CU2Z1S 155563099 Ki = 8190 nM T00176 CUE2F7 155564869 Ki = 630 nM T00176 C5IBV6 155565604 Ki = 430 nM T00176 C0OKH6 155566162 Ki = 6600 nM T00176 C1XMI2 155566670 Ki = 260 nM T00176 CBI1S9 155567165 IC50 = 10300 nM T00176 C3QM1J 155568384 Ki = 1910 nM T00176 C5D8PE 155569182 IC50 = 7100 nM T00176 C8KE3W 155569673 Ki = 520 nM T00176 D01QKK 216345 Ki = 30 nM T00176 D07QJJ 289 IC50 > 100000 nM T00176 D08EMG 736083 IC50 = 175 nM T00176 D08YAF 44412124 Ki = 6670 nM T00176 D0C0TN 248986 Ki = 120 nM T00176 D0M2EM 4650 IC50 = 13900 nM T38284 D00STL 644241 IC50 = 12.7 nM T38284 D0AZ3C 5291 IC50 = 14 nM T38284 D0E6XR 3062316 EC50 = 0.04 nM T38284 D0H0EQ 24826799 EC50 = 0.05 nM T38284 D0OB0F 5328940 IC50 = 20 nM T38284 D0R0MW 5329102 EC50 > 1000 nM T38284 D02LJW 23635314 IC50 = 100 nM T38284 D02XNW 5494449 IC50 = 50.12 nM T38284 D06JHV 46848036 IC50 = 6.2 nM T38284 D0E3TC 44259 IC50 = 121.8 nM T38284 D0U3EP 445154 IC50 = 28000 nM T38284 D05HDJ 49782106 EC50 = 7150 nM T38284 D0EF5T 44129660 EC50 = 430 nM T38284 D0JY1I 42613483 IC50 = 2700 nM T38284 D0L7XM 42628828 EC50 = 40 nM T38284 D0OE4F 4369496 IC50 = 100 nM T38284 D0ZH4I 76071870 IC50 > 10000 nM T38284 D01EFO 9864718 IC50 = 398.11 nM T38284 C6SB2N 123596 EC50 = 90 nM T38284 CV5MS2 2475277 EC50 = 1300 nM T38284 CCPF82 5312285 EC50 = 720 nM T38284 CZR3M4 9799152 IC50 = 100000 nM T38284 CY3MK1 9807952 IC50 = 3.981 nM T38284 CI3O6X 9814609 IC50 = 61659.5 nM T38284 CX9DG5 9822042 IC50 = 199.53 nM T38284 CSH0A9 9847014 IC50 = 346.74 nM T38284 C3UQL7 9860872 IC50 = 33884.42 nM T38284 CC90FJ 9869737 IC50 = 512 nM T38284 CIZ13L 9943193 IC50 = 602.56 nM T38284 CUKH27 9943194 IC50 = 707.95 nM T38284 CU78NO 9947433 IC50 = 151.36 nM T38284 CYT7R9 9953676 IC50 = 794.33 nM T38284 CJ40GO 9965429 IC50 = 1513.56 nM T38284 CTE3K0 9982070 IC50 = 3162.28 nM T38284 CP23QA 10007129 IC50 = 10 nM T38284 CLI9A3 10029363 IC50 = 63.1 nM T38284 C0G5DK 10039959 IC50 = 7943.28 nM T38284 CT9F2H 10053560 IC50 = 5.012 nM T38284 C8EW6P 10095381 IC50 = 2187.76 nM T38284 C3P8WK 10110378 IC50 = 1000 nM T38284 C63CFD 10111108 IC50 = 1288.25 nM T38284 CL42XS 10136330 IC50 = 794.33 nM T38284 CUW34X 10157645 IC50 = 1905.46 nM T38284 COC30E 10181160 IC50 = 199.53 nM T38284 CN51JQ 10292737 IC50 = 446.68 nM T38284 CG2L4Z 10343860 IC50 = 602.56 nM T38284 CYW13A 10348904 IC50 = 10 nM T38284 C7TJ9U 10483163 IC50 = 7.079 nM T38284 CS0DE8 10493971 IC50 > 3000 nM T38284 C78FPR 10501266 IC50 = 371.54 nM T38284 CU6G5Y 10708835 IC50 = 1202.26 nM T38284 CO61VZ 11161166 IC50 = 24000 nM T38284 C94MLD 11165739 EC50 = 390 nM T38284 C2KT9E 11168002 IC50 = 4.074 nM T38284 C89EZO 11180525 IC50 = 16.98 nM T38284 C3FL9M 11199480 IC50 > 100000 nM T38284 CJTP13 11280103 IC50 = 3801.89 nM T38284 CPW2Y8 11326963 EC50 = 4470 nM T38284 C1DF5Z 11336923 EC50 = 330 nM T38284 CKY3E2 11338122 IC50 = 199.53 nM T38284 CH4O8K 11347791 EC50 = 1660 nM T38284 C4RLW0 11368874 IC50 = 26000 nM T38284 C3OCV2 11371778 IC50 = 1000 nM T38284 CHJV86 11381980 EC50 = 470 nM T38284 C14XYD 11385486 IC50 > 10000 nM T38284 C3O0WI 11438191 IC50 = 5128.61 nM T38284 C3EXM4 11440028 IC50 = 398.11 nM T38284 C2E0GS 11461932 EC50 = 1800 nM T38284 C7I6AG 11474111 IC50 = 501.19 nM T38284 C0YH2X 11478363 IC50 = 1.25 nM T38284 CMW72Q 11488124 IC50 = 724.44 nM T38284 C57TKI 11565665 IC50 = 18000 nM T38284 C43JZU 11604436 IC50 = 3800 nM T38284 CGU7N0 11604739 IC50 = 12900 nM T38284 CLJ81E 11630507 IC50 = 20000 nM T38284 C6SGF3 11644985 IC50 = 16000 nM T38284 CJK78Z 11652152 IC50 = 8000 nM T38284 CAJS96 11662893 IC50 = 14600 nM T38284 CH3S9K 11666294 IC50 = 20000 nM T38284 C95EPO 11666668 IC50 = 35000 nM T38284 CKAH36 11669784 IC50 = 9500 nM T38284 CJ89UZ 11687939 IC50 > 100000 nM T38284 C7RDH3 11709536 IC50 > 100000 nM T38284 CFJ4I7 11723151 IC50 = 3311.31 nM T38284 C7C2FM 11737638 IC50 = 1513.56 nM T38284 CVFS29 11751305 IC50 = 64.57 nM T38284 CPJ7C9 11774222 EC50 = 580 nM T38284 CUDO23 11994441 IC50 = 25.12 nM T38284 C02DIH 14347011 IC50 = 1819.7 nM T38284 CZB2V0 16750146 IC50 = 20.89 nM T38284 C6XC2W 23145852 IC50 = 10.96 nM T38284 CUVB29 23145858 IC50 = 3.981 nM T38284 CO0T3M 24825778 IC50 = 750 nM T38284 CIFO50 24897305 IC50 = 11000 nM T38284 CYXC26 24958918 IC50 = 10000 nM T38284 CVUK27 24958920 IC50 = 2500 nM T38284 C35LZO 24959284 IC50 = 2500 nM T38284 CIZQ04 24959285 IC50 = 15000 nM T38284 C47ING 24959648 IC50 = 10000 nM T38284 C4V9GI 24960018 IC50 = 500 nM T38284 CWLR85 24960379 IC50 = 10000 nM T38284 CHC6A5 25017304 IC50 = 1378 nM T38284 C38YMD 25017555 IC50 = 7083 nM T38284 CDHM05 25017557 IC50 = 739.5 nM T38284 CFU60Y 25235817 IC50 = 436 nM T38284 C8B6TY 42628503 EC50 < 500 nM T38284 C15OSL 42633116 EC50 = 250 nM T38284 CO1I2D 42633117 EC50 = 1200 nM T38284 CO7YL0 42633119 EC50 > 10000 nM T38284 CWF2S8 42633305 EC50 = 160 nM T38284 CKCO80 42633306 EC50 = 400 nM T38284 CCI8P7 42633666 EC50 = 1320 nM T38284 CSH3I9 42633667 EC50 = 2200 nM T38284 CPNK96 42633668 EC50 = 4340 nM T38284 CL04QK 42633670 EC50 > 10000 nM T38284 C7DA0B 42633859 EC50 = 9680 nM T38284 CLM7B9 42634040 EC50 = 490 nM T38284 C6DK1W 42634389 EC50 > 10000 nM T38284 C87GKI 42634390 EC50 = 918 nM T38284 CK15FQ 42634392 EC50 = 406 nM T38284 CCN5O4 42634553 EC50 = 1340 nM T38284 C2H1SJ 42634556 EC50 = 48 nM T38284 C1M8SR 42634557 EC50 = 1960 nM T38284 C48YFI 42634730 EC50 = 5600 nM T38284 C8L5RN 42635093 EC50 = 150 nM T38284 CQ9F8I 42635272 EC50 = 120 nM T38284 CG2P1M 42635644 EC50 = 1230 nM T38284 C4JRG0 42635811 EC50 = 140 nM T38284 CCOV80 42635815 EC50 = 100 nM T38284 C7K9YE 44194683 EC50 = 420 nM T38284 C9G6QE 44194684 EC50 = 340 nM T38284 CBP7D2 44194685 EC50 = 240 nM T38284 CBD90A 44194780 EC50 = 920 nM T38284 COK3J5 44194781 EC50 = 970 nM T38284 C7XOD2 44194782 EC50 = 1150 nM T38284 C4T0HN 44194783 EC50 = 1270 nM T38284 C63UIZ 44194784 EC50 = 1240 nM T38284 CMRX16 44273620 IC50 = 5754.4 nM T38284 CCH89M 44300026 IC50 = 1995.26 nM T38284 CH4ND7 44340691 IC50 = 9772.37 nM T38284 CK2CU3 44340703 IC50 = 17378.01 nM T38284 CY0XF5 44340726 IC50 = 67608.3 nM T38284 C2F7SL 44395745 IC50 = 10000 nM T38284 C0TED6 44395746 IC50 = 5011.87 nM T38284 CZR42M 44395763 IC50 = 575.44 nM T38284 CJ0Z5K 44395813 IC50 = 8912.51 nM T38284 CU9XQ0 44395880 IC50 = 10000 nM T38284 CYF8U6 44395904 IC50 = 1000 nM T38284 C5DR6W 44395926 IC50 = 10000 nM T38284 C4R8EB 44410932 IC50 = 23000 nM T38284 CI82UE 45270897 IC50 > 10000 nM T38284 C4UM6Y 45273507 IC50 > 10000 nM T38284 CR4A6B 46703970 EC50 > 10000 nM T38284 CH9AW2 46865999 IC50 = 500 nM T38284 C4FX6S 46866098 IC50 = 500 nM T38284 CK6UL0 46866099 IC50 = 200 nM T38284 C67UEP 46881960 IC50 = 8 nM T38284 C71XDW 49780994 EC50 = 330 nM T38284 CEAH78 49780998 EC50 = 5000 nM T38284 CHS50Y 49780999 EC50 = 2920 nM T38284 C9WOE2 49781000 EC50 = 480 nM T38284 CGV34K 49781215 EC50 = 90 nM T38284 C84ZOI 49781216 EC50 = 360 nM T38284 C4K9DH 49781217 EC50 = 810 nM T38284 C34JPY 49781218 EC50 = 400 nM T38284 C7YET3 49781219 EC50 = 290 nM T38284 C48NTZ 49781220 EC50 = 170 nM T38284 C7QON3 49781221 EC50 > 10000 nM T38284 CHUG72 49781431 EC50 > 10000 nM T38284 CQ43VM 49781432 EC50 > 10000 nM T38284 CDU34O 49781433 EC50 > 10000 nM T38284 CSE62H 49781434 EC50 > 10000 nM T38284 CL51PM 49781435 EC50 > 10000 nM T38284 CE1N9P 49781436 EC50 > 10000 nM T38284 CF4TU7 49781437 EC50 > 10000 nM T38284 CH4MI1 49781662 EC50 > 10000 nM T38284 CQOW70 49781663 EC50 > 10000 nM T38284 C46TMR 49781664 EC50 > 10000 nM T38284 CG2I3L 49781665 EC50 > 10000 nM T38284 COW0H6 49781667 EC50 > 10000 nM T38284 CBH02L 49781668 EC50 = 1440 nM T38284 C6-DEC-09 49781877 EC50 > 10000 nM T38284 CGI64U 49781878 EC50 = 6890 nM T38284 C38FVM 49781879 EC50 = 380 nM T38284 CVT73X 49781880 EC50 = 760 nM T38284 C7X9UG 49781881 EC50 = 300 nM T38284 C5I3OF 49781882 EC50 = 270 nM T38284 C1T6CN 49782104 EC50 = 400 nM T38284 C6WOK4 49782105 EC50 = 350 nM T38284 CKQC50 49782107 EC50 = 6890 nM T38284 CWHY47 49782108 EC50 = 690 nM T38284 CGC82O 49782109 EC50 = 2960 nM T38284 C80XEK 49782334 EC50 = 6920 nM T38284 C2BNW5 49782337 EC50 = 160 nM T38284 C1EA9K 49782338 EC50 = 1700 nM T38284 C2Y6QS 50938552 IC50 > 10000 nM T38284 CS3LT9 51030149 IC50 = 671 nM T38284 C1XRG0 51030150 IC50 = 507 nM T38284 C3PDJ8 51030250 IC50 = 774 nM T38284 CAQ4V6 51030532 IC50 = 480 nM T38284 CX47EM 51030534 IC50 = 1300 nM T38284 CSZ36G 51030713 IC50 = 177 nM T38284 CA6U5X 51030714 IC50 = 491 nM T38284 C9NYP4 51036677 IC50 > 10000 nM T38284 C4WRY3 51037112 IC50 > 10000 nM T38284 CNWO03 51037408 IC50 = 5 nM T38284 CLO1I6 51037410 IC50 = 6 nM T38284 CZ2H3T 51037608 IC50 = 19 nM T38284 CK8J5T 51037609 IC50 = 904 nM T38284 CYO9W0 51037823 IC50 = 458 nM T38284 CF7HX6 51037824 IC50 = 161 nM T38284 CMX3I7 51037825 IC50 = 19 nM T38284 CRI28Z 51037948 IC50 > 10000 nM T38284 C4XT7P 51038497 IC50 = 24 nM T38284 CKB79R 51038498 IC50 = 125 nM T38284 C75JSI 51038499 IC50 = 7 nM T38284 C6PG5F 51351510 IC50 = 20.1 nM T38284 CHAV48 52940594 IC50 = 2500 nM T38284 CAK80G 52940928 IC50 = 2500 nM T38284 C02ALP 52940992 IC50 > 20000 nM T38284 CSM30J 52941799 IC50 = 2500 nM T38284 CFY5K7 52941942 IC50 = 10000 nM T38284 CPU53W 52941997 IC50 = 2500 nM T38284 C1LN4J 52942048 IC50 = 500 nM T38284 C69VKZ 52942052 IC50 = 2500 nM T38284 C0QFI8 52942203 IC50 > 20000 nM T38284 C7D5FE 52942236 IC50 > 20000 nM T38284 C0S7OM 52943049 IC50 = 2500 nM T38284 CQZ98C 52943259 IC50 = 2500 nM T38284 CZ3X7O 52943392 IC50 > 20000 nM T38284 C9L3HD 52943395 IC50 = 20000 nM T38284 CCBA25 52944595 IC50 > 20000 nM T38284 C1XN6P 52944599 IC50 > 20000 nM T38284 C1H8GZ 52944627 IC50 > 20000 nM T38284 C90JQR 52945824 IC50 > 20000 nM T38284 CPVD21 52945847 IC50 > 20000 nM T38284 C62EXZ 52946812 IC50 = 10000 nM T38284 C3WI7B 52947902 IC50 = 2500 nM T38284 CK08IW 52948022 IC50 = 2500 nM T38284 CJ1XR3 52948871 EC50 > 10000 nM T38284 C4Q6XB 52949498 IC50 > 20000 nM T38284 CCXY64 54581006 IC50 = 5510 nM T38284 C36DEH 54582045 IC50 = 277 nM T38284 CPI87W 54583990 IC50 > 2000 nM T38284 CIE67G 54585892 IC50 = 3780 nM T38284 CAIO65 68796885 EC50 = 0.04 nM T38284 C91HPI 71300299 IC50 > 5000 nM T38284 CC98EU 71449991 IC50 = 2.67 nM T38284 CV21PC 71449992 IC50 = 5.96 nM T38284 CG59TB 71449993 IC50 = 0.45 nM T38284 C23ETA 71450038 IC50 = 1.66 nM T38284 C3B7IP 71450039 IC50 = 0.36 nM T38284 C0XL6Z 71451816 IC50 = 2.25 nM T38284 CQM05U 71451817 IC50 = 0.6 nM T38284 CVE9P2 71451818 IC50 = 0.52 nM T38284 C30FHU 71453635 IC50 = 0.54 nM T38284 CR7DI8 71453636 IC50 = 1.01 nM T38284 C8K6BL 71453637 IC50 = 19.1 nM T38284 C12IUO 71453638 IC50 = 0.52 nM T38284 CIEK84 71453639 IC50 = 0.72 nM T38284 C0FTX4 71453675 IC50 = 0.33 nM T38284 CK7V6O 71453676 IC50 = 0.42 nM T38284 CU42QX 71455363 IC50 = 0.52 nM T38284 C4X9GT 71455364 IC50 = 0.78 nM T38284 CVY26H 71455365 IC50 = 1.18 nM T38284 C3X1OP 71455406 IC50 = 0.52 nM T38284 COUR46 71455407 IC50 = 1.03 nM T38284 C8IV0R 71455408 IC50 = 1.01 nM T38284 CY2G7S 71457180 IC50 = 0.7 nM T38284 CXA9W8 71457181 IC50 = 0.98 nM T38284 CCT0X3 71459003 IC50 = 17.8 nM T38284 C01XBA 71459004 IC50 = 2.56 nM T38284 C0WF3X 71459043 IC50 = 1.94 nM T38284 CJ3PO5 71459044 IC50 = 15 nM T38284 CW0X4B 71460798 IC50 = 3.44 nM T38284 CE84WT 71460799 IC50 = 12.8 nM T38284 CG0F1R 71460800 IC50 = 1629 nM T38284 CZM79U 71460801 IC50 = 22.6 nM T38284 CWT1E8 71460802 IC50 = 0.69 nM T38284 CZ72YB 71460803 IC50 = 302 nM T38284 C8KL1P 71460845 IC50 = 1.42 nM T38284 C7XZ6K 71460846 IC50 = 66 nM T38284 CS08OH 71462551 IC50 = 0.45 nM T38284 CB45LP 71462552 IC50 = 0.41 nM T38284 C1IT5U 71550931 IC50 = 355 nM T38284 C5V8IC 71602940 IC50 = 4.73 nM T38284 C6SV9J 71602987 IC50 = 4125.31 nM T38284 CCQ25W 71602988 IC50 = 4.79 nM T38284 C6LKO2 71602989 IC50 = 3.21 nM T38284 C93MLS 71602992 IC50 = 34.77 nM T38284 CSP7K1 71603051 IC50 = 2754.9 nM T38284 CH7D8G 71603053 IC50 = 3.78 nM T38284 CHZ7U8 71603054 IC50 = 294.34 nM T38284 CWE69D 71603113 IC50 = 0.52 nM T38284 C4WT7O 71603114 IC50 = 2.34 nM T38284 CR08FQ 71603115 IC50 = 1.48 nM T38284 CE09DT 71603116 IC50 = 350.08 nM T38284 C4NM3G 71603117 IC50 = 1110.42 nM T38284 C62ZYM 71603170 IC50 = 63.31 nM T38284 CU8Z1W 71603171 IC50 = 6.34 nM T38284 CG80HO 73345816 IC50 = 199.53 nM T38284 CKA92Y 73348812 IC50 = 33189.45 nM T38284 CEUP75 73351906 IC50 = 50118.72 nM T38284 C7DSE2 73351907 IC50 = 10000 nM T38284 C8SUY0 73354884 IC50 = 398.11 nM T38284 CPJC10 73356444 IC50 = 1000 nM T38284 CCIS39 73356445 IC50 = 5370.32 nM T38284 C2PAK9 73438493 IC50 = 10 nM T38284 CHI51J 76070594 IC50 = 390 nM T38284 C8VAD5 76070929 IC50 > 10000 nM T38284 CB4V1R 76071142 IC50 = 380 nM T38284 CBAT06 76071144 IC50 = 89 nM T38284 C7SH1T 76071506 IC50 = 210 nM T38284 CS87EI 76071624 IC50 = 880 nM T38284 CGC0K4 76071869 IC50 > 10000 nM T38284 C9A8IG 79072608 IC50 = 255 nM T38284 CBP5K7 91183030 IC50 > 10000 nM T38284 CO07DQ 101879028 IC50 = 50 nM T38284 CG7YK9 101879029 IC50 = 17 nM T38284 CS8N1X 101879030 IC50 = 130 nM T38284 CUSN35 101879031 IC50 = 70 nM T38284 CY7BI2 118706214 IC50 > 10000 nM T38284 CDIA30 118722069 IC50 = 78600 nM T38284 C2SFD8 118722070 IC50 = 354000 nM T38284 C7CKE4 118722071 IC50 > 500000 nM T38284 C9ZW4S 118722072 IC50 = 385 nM T38284 CJPC58 118722073 IC50 > 500000 nM T38284 C53MDX 118722074 IC50 = 141000 nM T38284 CFC4T9 118722075 IC50 > 500000 nM T38284 CO9AY0 118722076 IC50 = 16100 nM T38284 C7YB8R 118722077 IC50 > 500000 nM T38284 CHD5Y4 118722078 IC50 = 6060 nM T38284 CIQ5K8 118722079 IC50 = 1440 nM T38284 C6CW9X 118722080 IC50 = 13500 nM T38284 C0M1KE 118722081 IC50 = 872 nM T38284 C5TD1S 118722083 IC50 = 277000 nM T38284 CF3YQ1 118722084 IC50 > 500000 nM T38284 CPR97Z 118722085 IC50 > 500000 nM T38284 CZ0I1M 118722086 IC50 = 91800 nM T38284 C2ACT5 118722089 IC50 > 500000 nM T38284 C5LBT6 118722090 IC50 = 563 nM T38284 CQ1S2N 118722091 IC50 = 266000 nM T38284 CQCX41 118737057 IC50 = 1 nM T38284 CUP4S1 122183740 IC50 = 14.2 nM T38284 CT12MC 122183741 IC50 = 15.9 nM T38284 CV3FM4 122183742 IC50 = 213.5 nM T38284 CVM71G 122183743 IC50 = 41.02 nM T38284 C48MKU 122183744 IC50 = 43.27 nM T38284 C2MK8C 122183745 IC50 = 46.2 nM T38284 CN3VR2 122183746 IC50 = 50.6 nM T38284 C43ELH 122183747 IC50 = 178 nM T38284 CG71PU 122183748 IC50 = 326 nM T38284 CUWG02 122183749 IC50 = 129.1 nM T38284 C6SQI8 122183750 IC50 = 26.58 nM T38284 C5X8JH 122183808 IC50 = 117.4 nM T38284 CG3ZX6 122183809 IC50 = 16.87 nM T38284 CM3NO8 122183810 IC50 = 175.3 nM T38284 C2P9NG 122186622 IC50 > 1000 nM T38284 CSVT14 122186623 IC50 = 300 nM T38284 C2V7EG 122189041 IC50 > 500000 nM T38284 C6MU0Y 122189043 IC50 = 66 nM T38284 C19CBJ 122189044 IC50 = 1156 nM T38284 CEQ5W9 122189045 IC50 = 45600 nM T38284 C5EX7F 122189047 IC50 = 276 nM T38284 C0JYX4 122189048 IC50 = 60670 nM T38284 C4UK5I 122189049 IC50 = 10220 nM T38284 CDT8R6 122189050 IC50 = 112 nM T38284 CR2Y7P 122189051 IC50 = 63300 nM T38284 C5OR0G 122189052 IC50 = 940 nM T38284 C82CRO 122189053 IC50 > 500000 nM T38284 CJ9HI8 122189054 IC50 = 19070 nM T38284 C9JI1S 122189056 IC50 > 500000 nM T38284 CYF0W2 122189057 IC50 = 143 nM T38284 C2YT3F 122189058 IC50 > 500000 nM T38284 CDY7N9 122189059 IC50 = 5050 nM T38284 C9Y5NU 122189060 IC50 = 89700 nM T38284 C54KBN 122189061 IC50 = 73 nM T38284 CR81XY 122189062 IC50 = 321 nM T38284 C4NK6A 122189064 IC50 = 444180 nM T38284 CO36WE 122189065 IC50 = 16 nM T38284 CL72TM 122189066 IC50 = 421 nM T38284 C6ZHF0 122189067 IC50 = 1837 nM T38284 CQ2SD8 122189068 IC50 > 500000 nM T38284 CDX9H3 122190820 IC50 = 2590 nM T38284 CSV74J 122190821 IC50 = 8530 nM T38284 C3ZQJ4 122190822 IC50 = 14550 nM T38284 C4AM5V 122190823 IC50 > 100000 nM T38284 CU3O4Q 122190824 IC50 = 9250 nM T38284 C4BL5S 122190825 IC50 = 11300 nM T38284 CZBP91 122190826 IC50 = 9240 nM T38284 C3PB0Z 122190828 IC50 = 4400 nM T38284 CT32LN 122190829 IC50 = 6200 nM T38284 C1EBW9 122190830 IC50 = 8960 nM T38284 CZ26FY 122190831 IC50 = 73910 nM T38284 C5Z2DL 122190832 IC50 = 35660 nM T38284 CW84RP 122190867 IC50 > 100000 nM T38284 CHU8E2 122190868 IC50 = 42170 nM T38284 CF2W4A 122190869 IC50 = 35040 nM T38284 CUP8H1 122190870 IC50 = 15320 nM T38284 CFR2Z0 122190871 IC50 = 51920 nM T38284 CV2N9D 122190872 IC50 > 100000 nM T38284 CL42TR 122190873 IC50 > 100000 nM T38284 C6QY7L 122196083 IC50 = 14 nM T38284 CP0WN2 122196084 IC50 = 86 nM T38284 CG48DP 122196085 IC50 = 49200 nM T38284 C0LWG4 122196086 IC50 = 3410 nM T38284 C0I6AZ 122196188 IC50 = 180 nM T38284 CJCH07 122196189 IC50 > 100000 nM T38284 CM0X4J 122196190 IC50 = 2760 nM T38284 CA8U7J 122196191 IC50 = 83520 nM T38284 C8LAJ2 122196192 IC50 > 100000 nM T38284 C47IXK 122196193 IC50 = 2370 nM T38284 C6BPW7 122196194 IC50 = 1890 nM T38284 CFE6L4 122196195 IC50 = 22760 nM T38284 CN4J5W 122196196 IC50 = 8560 nM T38284 CI9J5Z 122196197 IC50 = 75290 nM T38284 CU9V8Q 122196198 IC50 = 31 nM T38284 CL07SV 122196199 IC50 = 18 nM T38284 CWU4J7 122196200 IC50 = 56270 nM T38284 CRXT48 122196201 IC50 > 100000 nM T38284 CEQ32S 122196202 IC50 = 250 nM T38284 CS3U0R 122196203 IC50 > 100000 nM T38284 CQL0W7 122197565 IC50 > 10000 nM T38284 C6KM3T 127034964 EC50 = 1 nM T38284 C1BZ4L 127034965 EC50 = 3 nM T38284 C3IRJ0 127048197 IC50 > 10000 nM T38284 CZ07TW 127048198 IC50 > 10000 nM T38284 CS0H2C 127048199 IC50 > 10000 nM T38284 C1OE2F 127049532 IC50 = 580 nM T38284 C5P8TC 127049857 IC50 > 10000 nM T38284 CPQ35R 127049870 IC50 = 3880 nM T38284 CQO3X7 127049871 IC50 > 10000 nM T38284 C5H8LK 127051998 IC50 > 10000 nM T38284 CGT0B1 127052321 IC50 > 10000 nM T38284 C7NH6A 127052914 IC50 > 10000 nM T38284 CKB1Y6 127052915 IC50 > 10000 nM T38284 C6RPF1 130364436 IC50 > 10000 nM T38284 CSY34O 130364443 IC50 > 10000 nM T38284 CI9H2W 130364450 IC50 > 10000 nM T38284 CM4TO5 130364451 IC50 = 2100 nM T38284 CV4DH7 130364460 IC50 > 10000 nM T38284 CW91ZV 130364461 IC50 > 10000 nM T38284 CQIZ43 130364463 IC50 = 9900 nM T38284 C4IKC6 130364464 IC50 > 10000 nM T38284 C0X6JS 130364465 IC50 > 10000 nM T38284 C0ZGC1 130364467 IC50 > 10000 nM T38284 CO9C5Q 130364468 IC50 > 10000 nM T38284 CQW3P1 130364471 IC50 > 10000 nM T38284 CHWX05 130364473 IC50 = 8700 nM T38284 CLB65Y 130364478 IC50 = 4300 nM T38284 CUZG19 130364481 IC50 > 10000 nM T38284 C34OMJ 130364482 IC50 > 10000 nM T38284 C6TWR3 130364484 IC50 > 10000 nM T38284 C8SF5Q 130364488 IC50 = 547 nM T38284 CS5C4E 130364494 IC50 > 10000 nM T38284 CVQ32Y 130364503 IC50 > 10000 nM T38284 CV8B0Y 130364506 IC50 > 10000 nM T38284 CHX23J 130364524 IC50 = 10000 nM T38284 CHYL89 130364535 IC50 > 10000 nM T38284 CBI35E 132275094 IC50 = 942 nM T38284 CCG06O 134131688 IC50 = 122000 nM T38284 CFE03W 134131725 IC50 = 16200 nM T38284 CC3Y5M 134131924 IC50 = 320 nM T38284 C60IDE 134134575 IC50 = 220 nM T38284 C4TJD6 134135198 IC50 = 24 nM T38284 CUP01F 134135273 IC50 = 19 nM T38284 CKQV02 134135339 IC50 > 500000 nM T38284 CM3J8P 134137546 IC50 = 58000 nM T38284 C9QFX5 134139856 IC50 = 2280 nM T38284 C6Q9BT 134140130 IC50 = 15 nM T38284 CF0M3H 134140636 IC50 = 2580 nM T38284 C4AI2O 134141645 IC50 = 0.012 ug.mL-1 T38284 C0UT6Y 134141669 IC50 > 500000 nM T38284 CZA63L 134143363 IC50 = 1980 nM T38284 C3NS0E 134144264 IC50 = 19 nM T38284 CEU0N9 134144345 IC50 = 1440 nM T38284 C0R1TX 134144394 IC50 = 640 nM T38284 CF7KV6 134144611 IC50 = 1150 nM T38284 C18KJH 134145016 IC50 = 0.012 ug.mL-1 T38284 C35XCY 134145509 IC50 = 1690 nM T38284 C7W6PG 134147256 IC50 = 4520 nM T38284 C8AJ9S 134148237 IC50 = 2250 nM T38284 CJ7A2M 134148351 IC50 = 440 nM T38284 C8YCR0 134148385 IC50 = 19 nM T38284 CCL1G8 134148410 IC50 = 2650 nM T38284 C37NPG 134148847 IC50 = 385 nM T38284 CUL93K 134150012 IC50 > 500000 nM T38284 CI4EO5 134150056 IC50 > 500000 nM T38284 C1EY7B 134153245 IC50 = 890 nM T38284 CLC89D 134153463 IC50 = 0.012 ug.mL-1 T38284 CFTL08 134155527 IC50 = 560 nM T38284 CAOK49 134155843 IC50 > 500000 nM T38284 CX6Q8G 134157397 IC50 > 500000 nM T38284 CQR94G 134198433 IC50 > 10000 nM T38284 C46QAS 135441185 EC50 = 10 nM T38284 C0PVG7 135819982 EC50 = 360 nM T38284 C2PJK6 135820173 EC50 = 70 nM T38284 C53LFX 135820297 EC50 = 970 nM T38284 CP7KZ8 135820466 EC50 = 1800 nM T38284 CQK62L 135820498 EC50 = 560 nM T38284 C4PD2G 135820511 EC50 = 30 nM T38284 CDT7E4 136211077 IC50 > 100 nM T38284 C5VE4K 137636547 IC50 > 10000 nM T38284 CZ05TY 137637593 IC50 > 10000 nM T38284 C6PKY7 137645383 IC50 > 10000 nM T38284 CHR9E0 137651685 IC50 = 414 nM T38284 CY53VO 137651787 IC50 > 10000 nM T38284 CE8DW7 137658399 IC50 > 10000 nM T38284 CU61WM 137658936 IC50 > 10000 nM T38284 CY9N8Q 137662234 IC50 = 8100 nM T38284 C0PYR1 138454771 EC50 < 10 nM T38284 CO9P7G 145351804 IC50 > 1000 nM T38284 CBR08X 145983359 IC50 = 1107 nM T38284 CE2X6V 145983518 IC50 = 435 nM T38284 C4ID8J 145984666 IC50 = 211 nM T38284 CD49VM 155295006 IC50 > 10000 nM T38284 CA8IF5 155510457 IC50 = 10660 nM T38284 CSHC63 155510467 IC50 > 10000 nM T38284 CG09WO 155512858 IC50 > 10000 nM T38284 C6H8ZU 155513172 IC50 = 2220 nM T38284 COI8N1 155513641 IC50 = 3720 nM T38284 CZDH58 155514096 IC50 > 10000 nM T38284 CEB08Z 155514919 IC50 = 6280 nM T38284 C84GJO 155517474 IC50 > 10000 nM T38284 CHQ5X7 155518340 IC50 = 6230 nM T38284 CP1B5K 155518600 IC50 = 520 nM T38284 C63PZX 155518871 IC50 > 10000 nM T38284 CC1A2U 155518947 IC50 = 4280 nM T38284 C1U3HE 155522045 IC50 = 110 nM T38284 C8EZ6J 155523550 IC50 = 31610 nM T38284 CF72IY 155527080 IC50 = 17560 nM T38284 CITV17 155527171 IC50 = 5750 nM T38284 C8DF2W 155529116 IC50 = 2160 nM T38284 CNP8T7 155530083 IC50 = 237 nM T38284 CK10UA 155531677 IC50 = 3696 nM T38284 C54ARD 155532371 IC50 = 170 nM T38284 C4DT6V 155532665 IC50 = 2340 nM T38284 CWLZ25 155535008 IC50 > 10000 nM T38284 C8NA6L 155536370 IC50 = 437 nM T38284 CL9X4S 155540971 IC50 = 2450 nM T38284 C3Q9UA 155541932 IC50 > 10000 nM T38284 CI27QV 155546853 IC50 > 10000 nM T38284 CYP2O5 155547984 IC50 = 1452 nM T38284 CB85AE 155550823 IC50 = 380 nM T38284 CL8KR2 155552517 IC50 = 989.3 nM T38284 C1TA9J 155553503 IC50 > 10000 nM T38284 CJS68O 155553593 IC50 = 290 nM T38284 C8BAU3 155554243 IC50 > 10000 nM T38284 CCQF25 155555943 IC50 > 10000 nM T38284 C9QM2K 155559937 IC50 = 1500 nM T38284 CN9LE6 155560662 IC50 = 5850 nM T38284 CHLY93 155562871 IC50 = 5345 nM T38284 C60KLJ 155564326 IC50 = 4992 nM T38284 C4BS6J 155565938 IC50 = 5637 nM T38284 CINX89 155566065 IC50 = 5120 nM T38284 CVMG35 155566307 IC50 = 1350 nM T38284 C7Q4RY 155566792 IC50 = 1813 nM T38284 CP69SU 155567937 IC50 > 10000 nM T38284 C8VT6Z 155568644 IC50 = 1990 nM T38284 D00AII 5281727 IC50 = 10000 nM T38284 D03EHM 24905142 IC50 = 18 nM T38284 D03NPX 447077 IC50 = 2 nM T38284 D03PLP 11579996 IC50 = 8000 nM T38284 D05UJT 5311510 EC50 = 140 nM T38284 D05XGZ 11536458 IC50 = 42000 nM T38284 D08RZB 11153014 IC50 = 3 nM T38284 D0AW4W 11537051 IC50 = 6000 nM T38284 D0AZ0Y 11514345 IC50 = 20000 nM T38284 D0H4YH 11594901 IC50 = 10000 nM T38284 D0I3XZ 11601743 IC50 = 4200 nM T38284 D0N7AJ 11409972 IC50 = 580 nM T38284 D0O9NE 5388063 IC50 = 10000 nM T38284 D0PI0R 11609210 IC50 = 14000 nM T38284 D0QG6G 11493254 IC50 = 14000 nM T72653 D0SN1T 456557 IC50 = 3200 nM T72653 C6AY2F 492577 IC50 = 8.95 nM T72653 CG03MO 492579 IC50 = 0.14 nM T72653 CU0J1O 492580 IC50 = 7.88 nM T72653 CG2YJ3 492581 IC50 = 213 nM T72653 CGT49R 492582 IC50 = 1031 nM T72653 C7YNV1 492583 IC50 = 13700 nM T72653 CU73IA 492587 IC50 = 0.76 nM T72653 CSM2C7 6476831 IC50 = 70.9 nM T72653 CVW1R8 6476832 IC50 = 2.77 nM T72653 C0YOX4 6476833 IC50 = 0.9 nM T72653 CN1S7G 6476834 IC50 = 0.68 nM T72653 CS5D8U 6476835 IC50 = 1.23 nM T72653 C2ZXI8 6476836 IC50 = 1.1 nM T72653 CTY56F 6476837 IC50 = 54 nM T72653 C4ELW7 6476838 IC50 = 775 nM T72653 CTWK35 6476839 IC50 = 391 nM T72653 CW4X1Q 6476840 IC50 = 13.2 nM T72653 CZ21FD 6477175 IC50 = 0.35 nM T72653 CL4A2K 9958342 Ki = 590 nM T72653 CPB2K3 44282128 IC50 = 3 nM T72653 C2N5AY 44282146 IC50 = 14.9 nM T72653 C7L6TW 44282191 IC50 = 16000 nM T72653 CRM3U9 44282585 IC50 = 12.3 nM T72653 CSY97P 44282615 IC50 = 7.22 nM T72653 CDE8J5 44282823 IC50 = 211000 nM T72653 CM0U2I 44282824 IC50 = 1000 nM T72653 CRZ2G6 44282840 IC50 > 350000 nM T72653 CLC1B6 44282841 IC50 = 12000 nM T72653 C2PQG1 44282987 IC50 = 70 nM T72653 C8FB5R 44282988 IC50 = 4500 nM T72653 C98IQA 56657646 Ki = 246000 nM T72653 CU8PH1 56661147 Ki = 11300 nM T72653 CIK1F8 56664602 Ki = 7150 nM T72653 CX73DJ 56671491 Ki = 1060000 nM T72653 CP43BU 56678250 Ki = 218000 nM T72653 CNP83W 56678251 Ki = 978000 nM T72653 CE67CG 56678252 Ki = 145000 nM T38179 D0QQ7D 123630 IC50 = 0.05 ug.mL-1 T38179 D0X7JN 5280980 IC50 = 0.005 ug.mL-1 T38179 C6O7YG 65754 IC50 = 0.013 ug.mL-1 T38179 CVU5J8 68118 IC50 = 1800000 ug.mL-1 T38179 CP1BV0 68146 IC50 = 33000 ug.mL-1 T38179 C90TYQ 130313 IC50 = 6500 nM T38179 C9BQ7M 10431019 IC50 = 200 nM T38179 CR5U8P 13056873 IC50 = 0.24 ug.mL-1 T38179 CQPY19 14556048 IC50 = 0.063 ug.mL-1 T38179 CN7Q8Y 23663400 IC50 = 290 nM T38179 CCT85Z 23682206 IC50 = 720 nM T38179 CL2G8U 23689319 IC50 = 0.54 ug.mL-1 T38179 C3A0EW 23690249 IC50 = 300 nM T38179 CQV82G 23697854 IC50 = 260 nM T38179 CFJ4L3 23714228 IC50 = 30 nM T38179 CXWM70 44264235 IC50 = 250 nM T38179 C8OSN5 44265260 IC50 = 34800 nM T38179 CY2C5N 44302976 IC50 = 640 nM T38179 C4NM5D 44302994 IC50 = 6760 nM T38179 C86QDI 44303012 IC50 = 44510 nM T38179 CFAZ65 44303014 IC50 = 527000 nM T38179 CJRV96 44303046 IC50 = 15.4 nM T38179 C6B9QS 44303048 IC50 = 1800 nM T38179 CNHM03 44303051 IC50 = 180 nM T38179 CQA6B4 44303062 IC50 = 310 nM T38179 CL82VY 44303065 IC50 = 196 nM T38179 CGEF89 44303072 IC50 = 9510 nM T38179 C8F6EZ 44303075 IC50 = 1 nM T38179 CWA0L5 44303141 IC50 = 592 nM T38179 C7BOX8 44303347 IC50 = 13200 nM T38179 C2O6NK 44303370 IC50 = 105 nM T38179 CH7X5U 44303373 IC50 = 26 nM T38179 CIO5V8 44303374 IC50 = 4 nM T38179 C8QMN5 44311630 IC50 = 0.04 ug.mL-1 T38179 CXLW39 44311932 IC50 = 0.2 ug.mL-1 T38179 C1PR7Y 44311943 IC50 = 0.16 ug.mL-1 T38179 CG2EH0 44311944 IC50 = 0.032 ug.mL-1 T38179 C5X0WF 44311970 IC50 = 0.05 ug.mL-1 T38179 CQPM39 44311971 IC50 = 0.1 ug.mL-1 T38179 CBY3D6 44311985 IC50 = 0.16 ug.mL-1 T38179 CYV9C0 44312261 IC50 = 0.05 ug.mL-1 T38179 C2EWL5 44312263 IC50 = 0.63 ug.mL-1 T38179 C0LX6K 44312264 IC50 = 0.13 ug.mL-1 T38179 C6O9MT 44312320 IC50 = 0.2 ug.mL-1 T38179 C0KHO4 44325415 IC50 = 0.36 ug.mL-1 T38179 C2JNG6 44325427 IC50 = 1 ug.mL-1 T38179 CSVJ16 44325596 IC50 = 0.014 ug.mL-1 T38179 C8GTV7 44325622 IC50 = 0.59 ug.mL-1 T38179 CRHI26 44325644 IC50 = 0.21 ug.mL-1 T38179 CY4I0R 44325660 IC50 = 0.0034 ug.mL-1 T38179 CH60RL 44377524 IC50 = 0.00055 ug.mL-1 T38179 C3BNW1 44380961 IC50 = 102000 nM T38179 CU61AD 44380999 IC50 = 932 nM T38179 C4TX7G 44381013 IC50 = 277000 nM T38179 CSD53W 44381030 IC50 = 230000 nM T38179 CF74JK 44381046 IC50 = 1130 nM T38179 CF7U4W 44381049 IC50 = 56500 nM T38179 CVCH40 44381110 IC50 = 844000 nM T38179 CAS43C 44381211 IC50 = 99200 nM T38179 C7I4WF 44381218 IC50 = 91100 nM T38179 CFW41B 44381342 IC50 = 173000 nM T38179 C0M4RO 44381438 IC50 = 100 nM T38179 CQJ9P0 44381472 IC50 = 31000 nM T38179 CHP68M 44381474 IC50 = 67000 nM T38179 C2L4XP 44381476 IC50 = 110000 nM T38179 CL6A2Z 44381483 IC50 = 240000 nM T38179 C1MX5A 44381487 IC50 = 75000 nM T38179 CWIT48 44381500 IC50 = 100000 nM T38179 CGPN35 44381504 IC50 = 1400 nM T38179 C3YDV5 44381537 IC50 = 4300 nM T38179 CLD9W8 44381589 IC50 = 7900 nM T38179 C4XQJ0 44381628 IC50 = 6000 nM T38179 CEKL21 44381631 IC50 = 33400 nM T38179 CD7L1R 44381779 IC50 = 15400 nM T38179 CRB03I 44381781 IC50 = 154000 nM T38179 CG7Q1B 44381784 IC50 = 280000 nM T38179 C1J8EA 44381801 IC50 = 8600 nM T38179 CLEW16 44381836 IC50 = 28000 nM T38179 CR5M7D 44381838 IC50 = 8900 nM T38179 CQRW20 76315023 IC50 = 0.065 ug.mL-1 T46628 D0H8VY 9853053 IC50 = 0.8 nM T46628 CC48GB 9805990 IC50 > 1000 nM T46628 CJ9NE6 9809160 IC50 = 14 nM T46628 CR8SJ9 9810471 IC50 = 9 nM T46628 CZB2L7 9827343 IC50 = 3.5 nM T46628 C5MQU2 9831128 IC50 < 10 nM T46628 CTP29B 9831229 IC50 = 12 nM T46628 CPV04O 9831585 IC50 = 3 nM T46628 C03LMO 9851010 IC50 = 180 nM T46628 C8GXC6 9853566 IC50 = 0.03 nM T46628 C2MJB3 9869236 IC50 = 70 nM T46628 CGS38K 9891662 IC50 = 204 nM T46628 C7OXU6 9893362 IC50 = 105 nM T46628 C95CAK 9893401 IC50 = 1000 nM T46628 CGQ63J 9912755 IC50 = 120 nM T46628 CV4W7Y 9917101 IC50 = 2.97 nM T46628 CQEU39 9940173 IC50 = 7 nM T46628 C7RW8K 9960070 IC50 = 11 nM T46628 CX47GA 10509221 IC50 = 1 nM T46628 CX4RE3 10557113 IC50 = 0.06 nM T46628 CDJ14F 10771201 IC50 = 0.24 nM T46628 C3OA2K 10771297 IC50 = 0.02 nM T46628 C8OX4Y 10818579 IC50 = 10 nM T46628 CA5FJ1 10842879 IC50 = 2 nM T46628 CO7JL9 10874540 IC50 = 90 nM T46628 CNQ27P 10875045 IC50 = 120 nM T46628 C3P9FZ 10895442 IC50 = 170 nM T46628 CC4SR0 10896240 IC50 = 34 nM T46628 C0GRI1 10896496 IC50 = 20 nM T46628 CRA54I 10917146 IC50 = 80 nM T46628 C57WJA 10918532 IC50 = 650 nM T46628 C6MJ3O 10928783 IC50 = 500 nM T46628 CK4O9I 10939283 IC50 = 100 nM T46628 CM9VK6 10939852 IC50 = 4800 nM T46628 CYU20M 10940136 IC50 = 120 nM T46628 C1IZR8 10951208 IC50 = 100 nM T46628 CVW5R3 10961434 IC50 = 110 nM T46628 CAHR01 10962353 IC50 = 100 nM T46628 CG8WC0 10962509 IC50 = 110 nM T46628 C62AUC 10973085 IC50 = 40 nM T46628 C1E3HD 10973138 IC50 = 240 nM T46628 CY7QP0 10983506 IC50 = 80 nM T46628 CN95OR 10983704 IC50 = 90 nM T46628 C96UMN 10994667 IC50 = 20 nM T46628 CN4QG3 10994772 IC50 = 50 nM T46628 COP90M 10995108 IC50 = 40 nM T46628 CIL7D4 10995390 IC50 = 20 nM T46628 C21TIL 11004943 IC50 = 100 nM T46628 C61DIZ 11027521 IC50 = 150 nM T46628 CX0I1A 11027680 IC50 = 80 nM T46628 CFVH36 11049142 IC50 = 70 nM T46628 CNE1M2 11123287 IC50 = 68 nM T46628 CQJR21 11124756 IC50 = 140 nM T46628 CSC8O9 11145136 IC50 = 70 nM T46628 CQEA84 11145472 IC50 = 70 nM T46628 CLE42U 11331363 IC50 = 0.0004 nM T46628 C4W1DI 11730355 IC50 = 710 nM T46628 CA9L4W 11733571 IC50 = 24 nM T46628 CLID72 11734494 IC50 = 14 nM T46628 C4LRQ2 11762346 IC50 = 80 nM T46628 CL4BI2 11762419 IC50 = 70 nM T46628 CQ9JC1 11827152 IC50 = 93 nM T46628 CWB17G 15603841 IC50 = 0.0028 nM T46628 CTYR34 16058735 IC50 > 10000 nM T46628 CCEJ98 16667090 IC50 > 10000 nM T46628 CU4IW5 16667135 IC50 > 10000 nM T46628 C3VF9Q 18409247 IC50 = 22 nM T46628 CZ1QO9 24797802 IC50 = 150 nM T46628 C38YMA 24999167 IC50 = 0.002 nM T46628 CY2R4C 25134625 IC50 = 710 nM T46628 CI6VC1 25211577 IC50 = 140 nM T46628 CJPE39 25211677 IC50 = 0.6 nM T46628 C1HO2U 44361523 IC50 = 170 nM T46628 CDZ19W 44361568 IC50 = 120 nM T46628 CBR57W 44361595 IC50 = 50 nM T46628 C4HPJ2 44361825 IC50 = 410 nM T46628 CHA20L 44361826 IC50 = 50 nM T46628 C2JC5G 44394851 IC50 = 9 nM T46628 CSZ1B9 44394967 IC50 = 5 nM T46628 CL93VZ 44411574 IC50 = 5.53 nM T46628 CRPC74 44411575 IC50 = 26.8 nM T46628 C3FMB2 44411576 IC50 = 29 nM T46628 C0TIF7 44411593 IC50 = 14.9 nM T46628 CG08PZ 44411594 IC50 = 13.29 nM T46628 CX4T6D 44411595 IC50 = 3.85 nM T46628 CY5OU8 44411596 IC50 = 6.38 nM T46628 CPQ9A4 44411597 IC50 = 1.64 nM T46628 CDV63C 44411601 IC50 = 72.7 nM T46628 CJN54C 44411611 IC50 = 85.5 nM T46628 C2LP6A 44411643 IC50 = 17.27 nM T46628 C5LRH6 44411644 IC50 = 35.92 nM T46628 CX71EU 44411645 IC50 > 100 nM T46628 CFC21A 44411646 IC50 > 100 nM T46628 C7WX5O 44411647 IC50 = 69.52 nM T46628 C5MNK6 44411655 IC50 = 4.11 nM T46628 C24BSY 44411656 IC50 = 1.75 nM T46628 C94CVR 44411657 IC50 = 3.5 nM T46628 COCB74 44411658 IC50 = 1.78 nM T46628 C6W1CY 44411678 IC50 = 15.6 nM T46628 C4H3YN 44411680 IC50 = 8.15 nM T46628 CL2A1V 44411681 IC50 = 5.05 nM T46628 CT2BE4 44411682 IC50 = 8.27 nM T46628 C87MVZ 44411684 IC50 > 100 nM T46628 C23FGJ 44411685 IC50 = 23.56 nM T46628 CGCN50 44411686 IC50 = 4.62 nM T46628 C84AST 44411696 IC50 = 96.71 nM T46628 CZY3C9 44411714 IC50 > 100 nM T46628 C4USD8 44411715 IC50 = 95.89 nM T46628 C8PA7T 44411734 IC50 = 29.51 nM T46628 CVTM68 44411735 IC50 = 69.39 nM T46628 C8BIS7 44411764 IC50 = 35.4 nM T46628 C4NQ1W 44411765 IC50 = 12.97 nM T46628 COUV59 44411780 IC50 = 2.34 nM T46628 C9HXE0 44411782 IC50 = 61.15 nM T46628 C2ZQY9 44411783 IC50 > 100 nM T46628 CV09DB 44411784 IC50 = 55.84 nM T46628 CJT6C8 44411785 IC50 > 100 nM T46628 C0QPN4 44411787 IC50 > 100 nM T46628 CZ5SY7 44411788 IC50 = 3.37 nM T46628 C9IRD1 44411833 IC50 = 23.13 nM T46628 CWH0O6 44411834 IC50 = 6.47 nM T46628 CFR5B9 44411845 IC50 = 1.68 nM T46628 CPAY94 44411848 IC50 = 5.28 nM T46628 C2CR4K 44411853 IC50 = 14.78 nM T46628 CL67IZ 44411854 IC50 = 7.14 nM T46628 C4BDL0 44411861 IC50 = 26.6 nM T46628 C2SG6R 44411862 IC50 = 17.38 nM T46628 CM0LK5 44411863 IC50 = 1.01 nM T46628 C4EHG5 44411872 IC50 = 5.67 nM T46628 CWC61A 44411873 IC50 = 11.78 nM T46628 CK9M4W 44411877 IC50 = 16.94 nM T46628 CKJ25X 44411881 IC50 > 100 nM T46628 CYI74K 44411882 IC50 = 69.84 nM T46628 CE2WQ3 44411883 IC50 > 100 nM T46628 C5BC4E 44411884 IC50 > 100 nM T46628 CX26GS 44411891 IC50 > 100 nM T46628 C91IKD 44411892 IC50 = 76.52 nM T46628 CP3Q5M 44411907 IC50 = 7.33 nM T46628 CC9Z0W 44411908 IC50 > 100 nM T46628 C85NDX 44411909 IC50 > 100 nM T46628 CA2T6I 44411910 IC50 = 9.43 nM T46628 C4HKM1 44411917 IC50 > 100 nM T46628 C2W1EC 44411948 IC50 = 22.46 nM T46628 CY16AU 44411949 IC50 = 18.3 nM T46628 CNW57Z 44411950 IC50 = 20.51 nM T46628 CJE9I0 44411971 IC50 = 13.27 nM T46628 CKTZ18 44411972 IC50 = 6.23 nM T46628 CJKS09 44411973 IC50 = 2 nM T46628 CG82NJ 44411978 IC50 = 16.93 nM T46628 C3N2SR 44411979 IC50 = 2.53 nM T46628 CRT70E 44591268 IC50 = 140 nM T46628 CVB19K 44591344 IC50 = 180 nM T46628 CPW59G 44591346 IC50 = 1400 nM T46628 CSM20Z 71449289 IC50 = 1.5 nM T46628 CE0B5Z 71449290 IC50 = 0.0095 nM T46628 C07UET 71449291 IC50 = 3 nM T46628 CFUV78 71449292 IC50 = 0.058 nM T46628 CUM3S9 71449293 IC50 = 0.021 nM T46628 CWFU91 71451082 IC50 = 2.8 nM T46628 CJ28HO 71451083 IC50 = 22 nM T46628 CE7P9A 71452903 IC50 = 0.55 nM T46628 CU1WH7 71452904 IC50 = 0.0007 nM T46628 CH8TC1 71452905 IC50 = 0.025 nM T46628 CQ49KJ 71452906 IC50 = 0.122 nM T46628 C8J6PN 71456408 IC50 = 0.378 nM T46628 C6WSN1 71456409 IC50 = 0.83 nM T46628 CIB4S3 71456410 IC50 = 0.066 nM T46628 C76QBL 71456411 IC50 = 0.253 nM T46628 C46CQK 71458256 IC50 = 0.001 nM T46628 C1BFR3 71458257 IC50 = 0.44 nM T46628 CNR6G8 71458258 IC50 = 0.101 nM T46628 CRD7U4 71460103 IC50 = 2.8 nM T46628 C8SQ7F 71460104 IC50 = 0.105 nM T46628 CD94LK 71460105 IC50 = 0.0074 nM T46628 CZ6N5M 71713624 IC50 = 33 nM T46628 CC9S1T 71713780 IC50 = 13 nM T46628 CM09QV 71713781 IC50 = 210 nM T46628 C8XR4A 71713782 IC50 = 25 nM T46628 CQS27Y 71713934 IC50 = 7 nM T46628 C21QNH 71713935 IC50 = 7400 nM T46628 D0J0TP 9917862 IC50 = 2.9 nM T70977 D04AIT 5280445 IC50 = 1500 nM T70977 D04LVK 57379345 IC50 > 10000 nM T70977 D07MGA 72281 IC50 = 26900 nM T70977 D0EG1I 9926791 IC50 > 10000 nM T70977 D0I9HF 10621 IC50 = 100000 nM T70977 D0J9ZR 4477 IC50 = 77500 nM T70977 D0K8KX 5280343 IC50 = 2000 nM T70977 D02RJY 11442891 IC50 > 10000 nM T70977 D02UFQ 11620908 IC50 > 10000 nM T70977 D03HUX 49792852 IC50 > 10000 nM T70977 D03LWG 53235510 IC50 > 10000 nM T70977 D05ADP 160355 IC50 = 130000 nM T70977 D05PZB 135398495 IC50 = 1 nM T70977 D06DMQ 59472121 Ki = 140 nM T70977 D07DTV 11338033 IC50 < 200 nM T70977 D07EHV 44814409 IC50 = 1300 nM T70977 D07HPJ 11476171 IC50 > 10000 nM T70977 D07SDQ 969516 IC50 = 17950 nM T70977 D08DHN 67286591 Ki = 1600 nM T70977 D0CY1B 6420138 Ki > 10000 nM T70977 D0E3TC 44259 IC50 = 4 nM T70977 D0H2HZ 60194098 IC50 = 5011.87 nM T70977 D0M0XB 10302451 IC50 > 10000 nM T70977 D0MS3Z 16725726 IC50 = 138 nM T70977 D0O0LS 25141092 IC50 > 10000 nM T70977 D0O6WV 24794418 IC50 > 2000 nM T70977 D0P1CV 46191454 IC50 = 79 nM T70977 D0Q9UX 16718576 IC50 > 10000 nM T70977 D0UT7X 11313622 IC50 = 78 nM T70977 D0Z1DH 10029385 IC50 = 0.9 nM T70977 D03BNU 59604787 IC50 > 10000 nM T70977 D0WS1V 448991 IC50 > 10000 nM T70977 D00OWF 5280953 IC50 > 10000 nM T70977 D00PWQ 3820 IC50 = 23 nM T70977 D06KNK 4124851 IC50 = 690 nM T70977 D09PGW 25253820 EC50 = 3200 nM T70977 D0A3MV 448014 IC50 = 2.07 nM T70977 D0N7BW 1276529 IC50 = 8990 nM T70977 D0NS6I 10037501 IC50 > 10000 nM T70977 D0Q3VZ 135398522 IC50 = 380 nM T70977 D0WX0K 71680628 Ki = 15 nM T70977 D0YK9D 9956119 IC50 = 30 nM T70977 D04FHB 6918852 Ki = 8000 nM T70977 D04WZK 10138980 Ki = 4.9 nM T70977 D09SFV 3973 IC50 = 8100 nM T70977 D0MC0O 135564570 IC50 = 31 nM T70977 D0R5ZR 127757 IC50 = 20 nM T70977 D0T3ME 156422 IC50 > 30000 nM T70977 CGAN35 2856 IC50 = 30 nM T70977 C6WUY3 3513 IC50 = 26 nM T70977 CQX7W5 4965 IC50 = 1000 nM T70977 CU7AC1 6259 IC50 = 5000 nM T70977 CV6BH8 6809 IC50 = 20220 nM T70977 CCW36T 7165 IC50 > 100000 nM T70977 CM0YU9 7364 IC50 > 100000 nM T70977 C7TZR4 7410 IC50 > 100000 nM T70977 CLZ46D 7454 IC50 = 500 nM T70977 C9A7WG 7467 IC50 > 100000 nM T70977 C97TNH 10177 IC50 = 4 nM T70977 C8IPB0 21639 IC50 = 100000 nM T70977 CYB5S8 23994 IC50 = 15000 nM T70977 C1MO0Y 28486 IC50 = 2000000 nM T70977 C6A7KB 49894 IC50 > 100000 nM T70977 CK2VX3 66840 IC50 = 2000 nM T70977 CV1X5G 67282 IC50 = 2500 nM T70977 CLA41H 68303 IC50 = 1000 nM T70977 CNUL24 69272 IC50 = 2500 nM T70977 CR42LP 70298 IC50 = 2500 nM T70977 C6T4QJ 75018 IC50 > 100000 nM T70977 CE9K5H 76052 IC50 > 100000 nM T70977 C8B7YP 98654 IC50 = 1500 nM T70977 C1P8WA 260652 IC50 > 10000 nM T70977 C6O5SK 280603 IC50 = 100000 nM T70977 C0DGC8 304747 IC50 > 10000 nM T70977 CL15BT 321979 IC50 = 5000 nM T70977 CD9XO4 326412 IC50 > 10000 nM T70977 CU4HI5 326413 IC50 > 10000 nM T70977 C6YML8 339916 IC50 = 2300 nM T70977 CG2V6U 343292 IC50 = 2456 nM T70977 CKC8L4 343879 IC50 > 100000 nM T70977 CZ9W0Y 356965 IC50 = 1690 nM T70977 C07MUW 366687 IC50 = 18230 nM T70977 CY26DN 369402 IC50 = 199.99 nM T70977 CMQE14 377824 IC50 = 2810 nM T70977 CID05G 381064 IC50 = 4700 nM T70977 CK9MS4 383434 IC50 = 113 nM T70977 C8QL0B 383785 IC50 = 23.99 nM T70977 CY3F2L 383786 IC50 = 199.99 nM T70977 C35EWT 383787 IC50 = 139.96 nM T70977 CX3A6O 384146 IC50 = 599.79 nM T70977 C09JHV 385068 IC50 = 2197.86 nM T70977 C9YCZ3 385069 IC50 = 130.02 nM T70977 CUYD71 385070 IC50 = 80 nM T70977 C06EVW 395169 IC50 = 4300 nM T70977 CDUC10 395170 IC50 = 119.95 nM T70977 CUL7P6 395804 IC50 = 799.83 nM T70977 CG0DM8 395805 IC50 = 100 nM T70977 CZX1J4 396079 IC50 = 30 nM T70977 C0RYZ9 396080 IC50 = 139958.73 nM T70977 CL0G3P 396081 IC50 = 899.5 nM T70977 C3HAR9 396411 IC50 = 15995.58 nM T70977 C7EN1O 396412 IC50 = 74.99 nM T70977 CC70DS 396571 IC50 = 1999.86 nM T70977 C0AZN2 396572 IC50 = 5000 nM T70977 CAE9J0 397216 IC50 = 10 nM T70977 CWIQ59 397718 IC50 = 500.03 nM T70977 CWSU67 397719 IC50 = 699.84 nM T70977 C5J1AF 398465 IC50 = 18 nM T70977 CGT4S0 400255 IC50 = 30000 nM T70977 C89SFG 400256 IC50 = 7200 nM T70977 CFBU18 400433 IC50 = 14810 nM T70977 C3K9FJ 401171 IC50 = 2500 nM T70977 CH20NR 403176 IC50 = 9 nM T70977 C3HX6M 406228 IC50 > 10000 nM T70977 CD9YQ6 406462 Ki = 14800 nM T70977 C7HME8 439246 IC50 = 45700 nM T70977 CB9F1O 447961 Ki = 20 nM T70977 C1ZG2U 449087 IC50 > 10000 nM T70977 CN8UJ7 520633 IC50 > 100000 nM T70977 CK57TY 563249 IC50 > 100000 nM T70977 CEY84H 580840 Ki = 460 nM T70977 C98MJC 582550 IC50 = 1500 nM T70977 CP9AM1 599038 Ki = 700 nM T70977 CE2G1Z 607858 Ki = 290 nM T70977 C96ZFR 624692 IC50 = 209 nM T70977 C6Y3ZP 626873 Ki = 23 nM T70977 CS9B3T 637482 IC50 = 11600 nM T70977 CO59EC 678545 IC50 > 100000 nM T70977 CU9Z0C 681957 IC50 = 5000 nM T70977 CQ7Z1F 682721 IC50 = 600 nM T70977 CN8SU3 684961 Ki = 1500 nM T70977 CPMJ63 707897 IC50 = 5960 nM T70977 C0FK8L 726568 IC50 = 338 nM T70977 CU9DG3 727529 IC50 > 10000 nM T70977 CZN6S9 743974 IC50 > 25118.86 nM T70977 C5LHO7 753058 Ki = 7300 nM T70977 C4AE2I 760516 IC50 = 214 nM T70977 CH7A2R 768611 IC50 = 8100 nM T70977 C14BYC 781209 IC50 = 2460 nM T70977 CQL20P 790035 IC50 > 10000 nM T70977 CXO42B 805390 IC50 = 1318 nM T70977 CXGH45 813164 IC50 > 100000 nM T70977 C53QBZ 837609 IC50 = 1291 nM T70977 CDSN72 838889 IC50 > 15000 nM T70977 CA1S6G 851256 IC50 = 12000 nM T70977 CQ1YV2 904180 IC50 = 917 nM T70977 CIW3E8 939111 IC50 = 17.2 nM T70977 CDRE31 963533 IC50 = 29000 nM T70977 CJ72IN 963534 IC50 = 235000 nM T70977 C0NF2R 1018252 IC50 = 11800 nM T70977 CU58RN 1048594 IC50 = 15790 nM T70977 C1Q4XB 1051604 IC50 = 862 nM T70977 CRK76I 1184346 IC50 = 1440 nM T70977 C7TH5J 1204987 IC50 > 10000 nM T70977 C6VCZ3 1205868 IC50 > 10000 nM T70977 C0SYZ7 1206234 IC50 > 10000 nM T70977 C02TQH 1224703 IC50 = 1150 nM T70977 CA0QI6 1227680 IC50 = 2495 nM T70977 C9Y0JC 1237187 IC50 > 10000 nM T70977 C2REL7 1239884 IC50 > 10000 nM T70977 C2JSX4 1241442 IC50 > 10000 nM T70977 CLC1U2 1270085 IC50 > 10000 nM T70977 C40DYT 1275119 IC50 = 8750 nM T70977 C6DYN7 1293837 IC50 = 12450 nM T70977 C9R8BJ 1350713 IC50 = 3970 nM T70977 CVJ8F0 1377751 IC50 > 10000 nM T70977 C1OW7H 1379703 IC50 > 10000 nM T70977 CIB51E 1379720 IC50 > 10000 nM T70977 CGM8O5 1398761 IC50 = 1420 nM T70977 CTV4Q6 1421105 IC50 = 7990 nM T70977 CA3GF2 1467927 IC50 = 10000 nM T70977 CU6EG0 1475221 Ki = 1490 nM T70977 CH9PR1 1547963 IC50 > 1000 nM T70977 C7ODT9 1550940 IC50 = 13700 nM T70977 CP42HJ 1625750 IC50 = 17000 nM T70977 C03SAD 1641793 IC50 > 10000 nM T70977 CA72ED 1724463 IC50 = 6900 nM T70977 CX23OE 1729742 IC50 > 100000 nM T70977 CX6SQ4 1749489 IC50 = 8750 nM T70977 CJ57GZ 1842529 IC50 = 3724 nM T70977 CRXA05 1988398 IC50 = 1000 nM T70977 C3PDL9 2079916 IC50 = 65 nM T70977 CH0Z5X 2131558 IC50 = 1100 nM T70977 COJ7W9 2134245 IC50 = 900 nM T70977 C2CT3B 2262763 IC50 = 5560 nM T70977 CE9ZN5 2291027 IC50 = 3570 nM T70977 C83QEW 2291265 IC50 = 2600 nM T70977 C5X7YV 2291327 IC50 = 2570 nM T70977 C29TYV 2673354 IC50 = 130 nM T70977 C1PXN0 2732733 IC50 = 2000 nM T70977 CW3G6T 2735867 IC50 = 1000 nM T70977 CX7S5O 2757188 IC50 = 10000 nM T70977 C29RQA 2757925 IC50 = 50000 nM T70977 C3ZI1K 2764173 IC50 = 23000 nM T70977 CG65XS 2764204 IC50 = 500 nM T70977 C82DNU 2795357 IC50 = 6000 nM T70977 CQ1Z5W 2797646 IC50 = 2500 nM T70977 CT5D7Y 2802986 IC50 > 10000 nM T70977 C1KPM5 3123256 IC50 = 13680 nM T70977 CZD5Q8 3132777 IC50 = 9600 nM T70977 CB0W9S 3242098 IC50 = 4000 nM T70977 CEAF95 3242308 IC50 > 100000 nM T70977 CT48FJ 3394376 IC50 = 4000 nM T70977 CNR0Z8 3882374 IC50 = 1231 nM T70977 CV84ZL 4145827 IC50 = 42700 nM T70977 CX4M8G 4153654 IC50 = 2800 nM T70977 CL4O0Z 4165708 IC50 = 50000 nM T70977 C6AE7U 4224626 IC50 > 100000 nM T70977 CV4JH9 4268708 IC50 > 10000 nM T70977 C0XR5L 4380991 IC50 = 830000 nM T70977 CH1D2N 4409556 IC50 = 3510 nM T70977 C25CJH 4596187 IC50 > 10000 nM T70977 CRL89Z 4613223 IC50 > 10000 nM T70977 C0I8LS 4663962 IC50 = 10.8 nM T70977 CORP43 4677904 IC50 = 10000 nM T70977 CG4E9X 4800452 IC50 > 1000 nM T70977 CI7BA0 4962248 IC50 > 100000 nM T70977 C6AD8F 5038004 Ki = 390 nM T70977 C2E6ZT 5101506 IC50 = 10000 nM T70977 C4ZA0C 5198245 IC50 = 2100 nM T70977 C7OWY4 5207527 IC50 > 10000 nM T70977 CU1N7T 5287990 IC50 = 40000 nM T70977 C54OLI 5288679 IC50 > 5000 nM T70977 C5K0BY 5324473 IC50 = 8390 nM T70977 CEJ0C2 5327664 IC50 = 35 nM T70977 CY6QK7 5327668 IC50 = 22 nM T70977 C0J4HV 5327709 IC50 = 90 nM T70977 C2E5SL 5327711 IC50 = 1.8 nM T70977 CSW8K7 5327715 IC50 = 3.6 nM T70977 CL5I2U 5330279 IC50 > 10000 nM T70977 C31FHN 5330788 IC50 > 20000 nM T70977 CG2VZ5 5331104 IC50 = 13 nM T70977 COFC04 5331105 IC50 = 33.04 nM T70977 C8WFJ1 5331108 IC50 = 199.99 nM T70977 CA4MH0 5331109 IC50 = 250.03 nM T70977 CNS20F 5331110 IC50 = 299.92 nM T70977 C6W0MJ 5331111 IC50 = 399.94 nM T70977 CR64JF 5331112 IC50 = 399.94 nM T70977 C1AN2V 5331115 IC50 = 349.95 nM T70977 CXF1P6 5331116 IC50 = 1199.5 nM T70977 CONC80 5331117 IC50 = 1399.59 nM T70977 CTNI84 5331118 IC50 = 1499.68 nM T70977 C1AV7M 5331119 IC50 = 1999.86 nM T70977 CE3XO1 5331120 IC50 = 1999.86 nM T70977 C5KP0C 5331121 IC50 = 2098.94 nM T70977 CELH01 5331122 IC50 = 2197.86 nM T70977 C9OW4Y 5331123 IC50 = 2301.44 nM T70977 CU6V3J 5331124 IC50 = 4000 nM T70977 CS4V6F 5331125 IC50 = 10000 nM T70977 CXK05J 5331126 IC50 = 23988.33 nM T70977 C7JM3R 5331128 IC50 = 179887.09 nM T70977 CB0PR6 5331131 IC50 = 639734.84 nM T70977 CLM7V5 5371900 IC50 = 14100 nM T70977 CZ1NX0 5384870 IC50 > 100000 nM T70977 CJD8Z3 5450091 IC50 = 6030 nM T70977 C9OL4F 5468481 IC50 = 4800 nM T70977 COR29P 5469423 IC50 = 15300 nM T70977 C5ZCB1 5469598 IC50 = 263 nM T70977 CZ03SJ 5476622 IC50 > 10000 nM T70977 CDK3J0 5703619 IC50 = 13 nM T70977 CK42AB 5708137 IC50 = 6010 nM T70977 CK7Y6A 5718019 IC50 = 584 nM T70977 CX5JO9 5793055 IC50 > 10000 nM T70977 CZLI06 5796182 IC50 = 4.19 nM T70977 CW1EK3 5881165 IC50 = 743 nM T70977 CW0V4C 5885463 IC50 > 10000 nM T70977 CA17GB 5892821 IC50 = 1560 nM T70977 C24TAU 5896893 IC50 > 10000 nM T70977 C3GS7L 5897747 IC50 > 10000 nM T70977 C7EMW0 5919090 IC50 = 218 nM T70977 CJR3H9 5928091 IC50 > 10000 nM T70977 C3SO9F 5961114 IC50 = 4200 nM T70977 CCXQ81 5983484 IC50 = 5540 nM T70977 CB2TY1 5998116 IC50 = 678 nM T70977 C5V0TR 6070143 IC50 > 10000 nM T70977 CG1JV6 6086375 IC50 = 18200 nM T70977 CT72OW 6115642 IC50 = 9220 nM T70977 C7PZV1 6249565 IC50 > 10000 nM T70977 CEZP52 6263849 IC50 = 250 nM T70977 C9AG1B 6538742 IC50 = 4197.59 nM T70977 CU7S1Y 6538743 IC50 = 1300.17 nM T70977 C9UE7W 6538744 IC50 = 239.88 nM T70977 C3WVA9 6538745 IC50 = 11994.99 nM T70977 CEB5H8 6538746 IC50 = 18 nM T70977 CA8XN6 6538749 IC50 = 89.95 nM T70977 C9GO5D 6538750 IC50 = 500034.53 nM T70977 CN63QP 6538751 IC50 = 5296.63 nM T70977 CSFM17 6538752 IC50 = 130.02 nM T70977 CY7RX2 6538753 IC50 = 69.98 nM T70977 C48XPN 6538754 IC50 = 21.98 nM T70977 C1SU7T 6538756 IC50 = 5495.41 nM T70977 CO97TH 6538757 IC50 = 599.79 nM T70977 CI3N9D 6538758 IC50 = 1000000 nM T70977 CHIA01 6538759 IC50 = 29.99 nM T70977 CRE5Z7 6538762 IC50 = 1300.17 nM T70977 CRC4Q1 6538763 IC50 = 399.94 nM T70977 CD8OK3 6538764 IC50 = 330.37 nM T70977 CAV08B 6538765 IC50 = 34.99 nM T70977 C9W8PB 6538766 IC50 = 3300 nM T70977 CGRW90 6538768 IC50 = 3200 nM T70977 CK3U1Q 6538770 IC50 = 1100 nM T70977 CHS28P 6538772 IC50 = 60000 nM T70977 CP30VA 6538773 IC50 = 85000 nM T70977 CZWH53 6538774 IC50 = 1900 nM T70977 C9ST0Q 6538776 IC50 > 100000 nM T70977 CN92BX 6538777 IC50 = 6000 nM T70977 CAB7F2 6538778 IC50 = 7200 nM T70977 CCD5J4 6538779 IC50 = 4800 nM T70977 CY7UA9 6538780 IC50 = 2600 nM T70977 CAY80Z 6538781 IC50 = 12000 nM T70977 C8NT0Z 6538782 IC50 = 460 nM T70977 CQ9J3G 6538783 IC50 = 2000 nM T70977 C5I6GK 6538784 IC50 = 400 nM T70977 C02GBE 6538785 IC50 = 2500 nM T70977 CW4DQ5 6538786 IC50 = 500 nM T70977 C4Z6WY 6538787 IC50 = 600 nM T70977 C8YKR3 6538788 IC50 > 10000 nM T70977 CN2WA5 6538789 IC50 = 1100 nM T70977 C2OXJ4 6538790 IC50 = 6800 nM T70977 C9AT4Z 6538791 IC50 = 500 nM T70977 CLH35K 6538792 IC50 = 1700 nM T70977 C8JAO7 6538793 IC50 = 750 nM T70977 C5ZR1B 6538794 IC50 = 5900 nM T70977 CD5C0A 6538795 IC50 = 6800 nM T70977 CWE3U0 6538796 IC50 = 1000 nM T70977 CMVJ20 6538797 IC50 = 8000 nM T70977 CA3IJ9 6538801 IC50 = 15000 nM T70977 CD5LE1 6538802 IC50 = 1200 nM T70977 CHER71 6538803 IC50 = 800 nM T70977 CE41TC 6538804 IC50 = 15000 nM T70977 C2IF9T 6538805 IC50 = 27000 nM T70977 CTW29F 6538806 IC50 > 100000 nM T70977 C16FEL 6538807 IC50 = 1000 nM T70977 C62LHV 6538808 IC50 = 18000 nM T70977 C3DM7P 6538809 IC50 = 20000 nM T70977 CYWL90 6538810 IC50 > 100000 nM T70977 CH13FR 6538884 IC50 = 530 nM T70977 C7YEI4 6538887 IC50 = 7360 nM T70977 C7C6AK 6538896 IC50 = 6000 nM T70977 C6PGU5 6539132 IC50 = 5000 nM T70977 C92ATH 6539133 IC50 = 25000 nM T70977 CXV16Y 6539134 IC50 = 10000 nM T70977 C19LGP 6539135 IC50 = 35000 nM T70977 CG1JC0 6539136 IC50 = 10000 nM T70977 CW1BY5 6539138 IC50 > 100000 nM T70977 C31HEX 6539139 IC50 = 7000 nM T70977 C9V2RS 6539140 IC50 = 10000 nM T70977 CM3U6H 6539141 IC50 = 3000 nM T70977 C1H9IL 6539142 IC50 = 4000 nM T70977 CDVA03 6539143 IC50 = 6000 nM T70977 CK5IP7 6539144 IC50 = 4000 nM T70977 CB8QX1 6539145 IC50 = 6000 nM T70977 CD60HP 6539146 IC50 = 5000 nM T70977 CMET61 6539147 IC50 = 2000 nM T70977 CO2S1F 6539148 IC50 = 3000 nM T70977 C9VQF2 6539149 IC50 = 20000 nM T70977 CH9W5T 6539150 IC50 = 8000 nM T70977 CO3NE8 6539151 IC50 = 6000 nM T70977 C1Q7CK 6539152 IC50 = 10000 nM T70977 C97MFS 6539154 IC50 = 65000 nM T70977 CQ5E2M 6539166 IC50 = 3000 nM T70977 CGS97O 6539167 IC50 = 25000 nM T70977 C5RCG8 6539168 IC50 = 1000 nM T70977 C1A6GX 6539169 IC50 = 2000 nM T70977 CNX9U0 6539170 IC50 = 1500 nM T70977 CVR1Z5 6539171 IC50 = 1000 nM T70977 CWA2U1 6539172 IC50 = 8000 nM T70977 CK2S4G 6539176 IC50 = 5000 nM T70977 C1AUO5 6539177 IC50 = 75000 nM T70977 C1F2ZR 6539178 IC50 > 100000 nM T70977 CWT15Z 6539179 IC50 = 5000 nM T70977 CM2N8O 6539359 Ki = 10 nM T70977 CTD0X9 6539360 Ki = 19900 nM T70977 CUK02R 6539362 IC50 = 5 nM T70977 CZY97M 6539363 IC50 = 5 nM T70977 C9X8DW 6539364 IC50 = 16 nM T70977 CM9FT4 6539365 Ki = 120 nM T70977 C9Y3KC 6539366 Ki = 50 nM T70977 C6Z0WU 6539368 Ki < 10 nM T70977 CY1W7D 6539369 IC50 = 1 nM T70977 CO3A4B 6539370 Ki = 10 nM T70977 C8RND3 6539371 Ki < 10 nM T70977 CB69DA 6539372 Ki = 10 nM T70977 CL18KE 6539373 Ki < 10 nM T70977 C74TAS 6539375 Ki < 10 nM T70977 C2GFT6 6539376 Ki < 10 nM T70977 C7SHN5 6539377 Ki < 10 nM T70977 CQM14U 6539378 Ki < 10 nM T70977 CTBE09 6539379 IC50 = 1 nM T70977 CWN7Q3 6539380 Ki = 10 nM T70977 CN2XV5 6539381 Ki = 50 nM T70977 C5TC2D 6539382 Ki = 190 nM T70977 C8KT3B 6539383 Ki = 790 nM T70977 CQ84MY 6539384 Ki = 100 nM T70977 C5Z4AQ 6539385 Ki = 50 nM T70977 CZQ56A 6539386 Ki = 50 nM T70977 CA5YC3 6539387 Ki = 70 nM T70977 C6A0FQ 6539388 Ki = 120 nM T70977 CX0T4J 6539389 Ki = 190 nM T70977 C7E2ZP 6539390 Ki = 3160 nM T70977 CAP2D7 6539391 Ki = 630 nM T70977 CYC62P 6539392 Ki = 30 nM T70977 C9NC7H 6539393 Ki < 10 nM T70977 C4R2HQ 6539394 Ki = 50 nM T70977 CU85HS 6539395 Ki = 10 nM T70977 CQ51SX 6539396 Ki = 10 nM T70977 CFVB56 6539397 Ki = 150 nM T70977 C8K7LC 6539398 Ki = 120 nM T70977 C6K7UA 6539399 Ki = 10 nM T70977 C5U4AD 6539400 Ki = 10 nM T70977 CO04SD 6539401 Ki = 10 nM T70977 CC0Q9Z 6539402 Ki = 10 nM T70977 C5S6FX 6539403 Ki = 20 nM T70977 CNR94M 6539404 Ki < 10 nM T70977 CVD04S 6539405 Ki = 20 nM T70977 C3BCG6 6539406 Ki = 20 nM T70977 CEV0Q5 6539407 Ki = 20 nM T70977 C9PRY5 6539408 Ki = 40 nM T70977 C1L3BI 6539409 Ki = 10 nM T70977 C72GAY 6539410 Ki = 5010 nM T70977 CZ67GY 6539411 Ki = 31600 nM T70977 C9G2CO 6539412 Ki = 7940 nM T70977 C9VEJ5 6539413 Ki = 31000 nM T70977 CF9AB1 6539414 Ki = 5010 nM T70977 C5TUV1 6539415 Ki > 31600 nM T70977 CCES70 6539416 Ki > 31600 nM T70977 CWAN68 6539417 Ki > 31600 nM T70977 CXI64Y 6539418 Ki > 31600 nM T70977 C97DXU 6539419 Ki > 31600 nM T70977 CO39EQ 6539420 Ki = 150 nM T70977 C7A1QZ 6539421 Ki = 310 nM T70977 CA04MW 6539422 Ki = 50 nM T70977 CG5ZY9 6539423 Ki = 1000 nM T70977 C92LYE 6539424 Ki = 1250 nM T70977 CU9A6K 6539425 Ki = 2510 nM T70977 C2FUA0 6539426 Ki = 1000 nM T70977 CD4Z7F 6539427 Ki = 3980 nM T70977 CG6C5K 6539428 Ki = 790 nM T70977 CPS9K1 6539429 Ki = 50 nM T70977 C9JW4Z 6539430 IC50 = 39.81 nM T70977 C6NW0F 6539431 Ki = 30 nM T70977 CK0MH3 6539432 Ki = 100 nM T70977 C35HXQ 6539433 Ki = 30 nM T70977 C0RS9Q 6539434 Ki = 790 nM T70977 CWZE47 6539435 Ki = 1580 nM T70977 CIRF95 6539436 Ki = 630 nM T70977 C6RIL5 6539437 Ki = 150 nM T70977 CCEB18 6539438 Ki > 31600 nM T70977 C9FRV1 6539439 Ki > 31600 nM T70977 CS1K9T 6539440 Ki = 20 nM T70977 CD26TN 6539441 Ki = 20 nM T70977 C6U4BK 6539442 Ki = 10 nM T70977 CPU3R1 6539443 Ki = 10 nM T70977 CP36QM 6539444 Ki = 50 nM T70977 CQ39BD 6539445 Ki = 19000 nM T70977 CJO9W0 6539446 Ki = 23000 nM T70977 C7X8AJ 6539447 Ki > 19950 nM T70977 C1LV4T 6539448 Ki > 19950 nM T70977 C7M9VJ 6539449 Ki = 80 nM T70977 CM8J1K 6539450 Ki = 6000 nM T70977 CV1EC6 6539452 IC50 = 216 nM T70977 C0MW6H 6539453 IC50 = 216 nM T70977 C95UNH 6539454 IC50 = 141 nM T70977 CHQB47 6539455 IC50 = 514 nM T70977 CK0QF7 6539456 IC50 = 390 nM T70977 CC2N8D 6539457 IC50 = 301 nM T70977 CO5ZI9 6539458 IC50 = 195 nM T70977 CUQ6F3 6539459 IC50 = 114 nM T70977 CD94GZ 6539460 IC50 = 104 nM T70977 CXI9R2 6539461 IC50 = 257 nM T70977 COG8F9 6539462 IC50 = 70 nM T70977 CSN2M8 6539463 IC50 = 447 nM T70977 C7G9QY 6539464 IC50 = 156 nM T70977 C09GEI 6539465 IC50 = 704 nM T70977 C4MA9R 6539466 IC50 = 374 nM T70977 C3B1MV 6539467 IC50 = 259 nM T70977 CZC31W 6539468 IC50 = 251 nM T70977 CC17FL 6539469 IC50 = 1478 nM T70977 CT8Z5A 6539470 IC50 = 472 nM T70977 CQ8P2W 6539471 IC50 = 236 nM T70977 C0CPN8 6539472 IC50 = 407 nM T70977 C7OFY0 6539473 IC50 = 481 nM T70977 CXQB76 6539474 IC50 = 123 nM T70977 CSYM79 6539475 IC50 = 317 nM T70977 CX1PB2 6539476 IC50 = 152 nM T70977 CD0MK5 6539477 IC50 = 139 nM T70977 C0V8PK 6539478 IC50 = 94 nM T70977 CW1FA4 6539479 IC50 = 59 nM T70977 CQT3S5 6539480 IC50 = 173 nM T70977 CMHO38 6539481 IC50 = 149 nM T70977 CRB06P 6539482 IC50 = 93 nM T70977 C0QV9A 6539483 IC50 = 82 nM T70977 CB1I5W 6539484 IC50 = 52 nM T70977 CO4EP0 6539485 IC50 = 58 nM T70977 C15YWK 6539486 IC50 = 142 nM T70977 CB01VH 6539487 IC50 = 20 nM T70977 CBZ2U6 6539488 IC50 = 91 nM T70977 C0CA1Y 6539489 IC50 = 83 nM T70977 C3ZF8P 6539490 IC50 = 71 nM T70977 CEI56T 6539491 IC50 = 291 nM T70977 CR3A6L 6539492 IC50 = 136 nM T70977 CT2H9L 6539493 IC50 = 134 nM T70977 C9LYZ2 6539494 IC50 = 195 nM T70977 C0ZDY3 6539495 IC50 = 79 nM T70977 CR72NT 6539496 IC50 = 186 nM T70977 C6DKW8 6539497 IC50 = 214 nM T70977 CD0T4H 6539498 IC50 = 143 nM T70977 CXS64M 6539499 IC50 = 74 nM T70977 CI2AZ0 6539500 IC50 = 28 nM T70977 C5YWB1 6539501 IC50 = 85 nM T70977 CX9V7E 6539502 IC50 = 109 nM T70977 CUWN19 6539503 IC50 = 404 nM T70977 C0P3JF 6539504 IC50 = 161 nM T70977 CG8Q3U 6539505 IC50 = 110 nM T70977 CM58CR 6539506 IC50 = 532 nM T70977 CN4JS2 6539507 IC50 = 203 nM T70977 CNE79Y 6539508 IC50 = 152 nM T70977 C3YRL2 6539509 IC50 = 529 nM T70977 CY5NZ6 6539510 IC50 = 243 nM T70977 CP86TH 6539511 IC50 = 392 nM T70977 C8D5RK 6539512 IC50 = 2613 nM T70977 C5T8YX 6539514 IC50 = 1398 nM T70977 C1K8EO 6539515 IC50 = 2285 nM T70977 CILQ58 6539516 IC50 = 337 nM T70977 CA9KF0 6539517 IC50 = 187 nM T70977 CLV36F 6539518 IC50 = 131 nM T70977 C37DQI 6539519 IC50 = 460 nM T70977 CX7A4E 6539520 IC50 = 161 nM T70977 CD4A1X 6539521 IC50 = 1412 nM T70977 CXS23C 6539522 IC50 = 694 nM T70977 C6R3GO 6539523 IC50 > 5000 nM T70977 CF3S6U 6539526 IC50 = 7 nM T70977 CG8ZC5 6539528 IC50 = 430 nM T70977 CVE25D 6539529 IC50 = 1260 nM T70977 CR7JG1 6539530 IC50 = 23000 nM T70977 C5J1RN 6539531 IC50 = 23000 nM T70977 C7RA9C 6539532 IC50 = 23000 nM T70977 C0GI9Y 6539533 IC50 = 291 nM T70977 CL54CB 6539534 IC50 = 43 nM T70977 C8ZTV0 6539535 IC50 = 56 nM T70977 CETM71 6539536 IC50 = 19 nM T70977 CKM15E 6539537 IC50 = 5 nM T70977 CFS2R3 6539538 IC50 = 2810 nM T70977 C31TYK 6539539 IC50 = 3572 nM T70977 C0MG7X 6539540 IC50 = 356 nM T70977 CP7SM9 6539541 IC50 = 2343 nM T70977 CX90YS 6539542 IC50 = 18 nM T70977 C63YHD 6539543 IC50 = 20 nM T70977 C8BD2P 6539544 IC50 = 7 nM T70977 CJI31S 6539545 IC50 = 27 nM T70977 CX6M9C 6539546 IC50 = 11 nM T70977 C3JBE0 6539547 IC50 = 443 nM T70977 C53JWE 6539548 IC50 = 851 nM T70977 C87EVK 6539549 IC50 = 169 nM T70977 CVGH07 6539550 IC50 = 241 nM T70977 CQ74FL 6539551 IC50 = 99 nM T70977 C5M3BE 6539552 IC50 = 2697 nM T70977 C9D1ME 6539553 IC50 = 691 nM T70977 CU61ZB 6539554 IC50 = 22 nM T70977 CL2RW0 6539555 IC50 = 11 nM T70977 C5SGK0 6539556 IC50 = 7 nM T70977 CXV5C7 6539557 IC50 = 5 nM T70977 C7L2OQ 6539558 IC50 = 9 nM T70977 CTU82J 6539559 IC50 = 5 nM T70977 CL20EZ 6539565 IC50 = 425 nM T70977 CMN15O 6539567 IC50 = 23000 nM T70977 CP7J3S 6539569 IC50 = 8 nM T70977 CS6T9C 6539570 IC50 = 125 nM T70977 C8B5SQ 6539572 IC50 = 1593 nM T70977 CC12VG 6539577 IC50 = 415 nM T70977 C7C9BO 6539578 IC50 = 75 nM T70977 CIT1W5 6539579 IC50 = 234 nM T70977 CVSZ60 6539580 IC50 = 87 nM T70977 C0V5BI 6539581 IC50 = 383 nM T70977 CX9V6S 6539585 IC50 = 21 nM T70977 CCXU69 6539586 IC50 = 215 nM T70977 CQTU34 6539587 IC50 = 329 nM T70977 COI57D 6539588 IC50 = 39 nM T70977 CQ97IV 6539591 IC50 = 7 nM T70977 C70OTV 6539592 IC50 = 141 nM T70977 CAI54V 6539593 IC50 = 498 nM T70977 C9ABL1 6539595 IC50 = 42 nM T70977 C4TJI2 6539598 IC50 = 481 nM T70977 C79LMV 6539603 IC50 = 1000 nM T70977 CNV39L 6539606 IC50 = 828 nM T70977 C14VJA 6539608 IC50 = 320 nM T70977 C7U2TC 6539610 IC50 = 35 nM T70977 C5XBK1 6539611 IC50 = 7 nM T70977 CNE0Y5 6539612 IC50 = 99 nM T70977 CK3W6M 6539613 IC50 = 16 nM T70977 C1PVJ8 6539615 IC50 = 14 nM T70977 CT5UI2 6539716 IC50 = 1200 nM T70977 C5Q8KG 6539717 IC50 = 11000 nM T70977 CFK8H1 6539718 IC50 = 8000 nM T70977 CP9D8T 6539727 IC50 > 250000 nM T70977 CDJB93 6539728 IC50 > 250000 nM T70977 C9H2LF 6539729 IC50 > 250000 nM T70977 CSUA12 6539730 IC50 = 29000 nM T70977 CZG72R 6539731 IC50 = 820 nM T70977 C1SOF9 6539733 IC50 = 198000 nM T70977 C7TQA0 6539734 IC50 = 1400 nM T70977 C1L0CM 6539735 IC50 = 1100 nM T70977 CLN13I 6539736 IC50 > 250000 nM T70977 CUM72Z 6539737 IC50 = 80 nM T70977 CNFV70 6539738 IC50 = 437 nM T70977 CBRC53 6539739 IC50 = 537 nM T70977 C8QG1T 6539740 IC50 = 130 nM T70977 CW7VD6 6539741 IC50 = 316 nM T70977 C5UFS1 6539742 IC50 = 30 nM T70977 C5XSJ6 6539743 IC50 = 320 nM T70977 CRL2P4 6539744 IC50 = 1820 nM T70977 CSWR78 6539745 IC50 > 34000 nM T70977 CXI8M7 6539746 IC50 = 1950 nM T70977 CSZF21 6539747 IC50 > 35000 nM T70977 CFM2K9 6539748 IC50 = 2400 nM T70977 C1QFC6 6539749 IC50 = 170 nM T70977 CFQ5R7 6539750 IC50 = 1000 nM T70977 C0R6WV 6539751 IC50 = 617 nM T70977 C25FMB 6539752 IC50 = 575 nM T70977 CRB1O3 6539753 IC50 = 5 nM T70977 CZ17AH 6539754 IC50 = 20 nM T70977 CT4K0Z 6539755 IC50 = 550 nM T70977 CMIS20 6539756 IC50 = 240 nM T70977 CTNR52 6539757 IC50 = 219 nM T70977 CJ58QK 6539758 IC50 = 5 nM T70977 CL9IM4 6877491 IC50 = 410 nM T70977 CVU8N0 6918710 IC50 = 1600 nM T70977 CS20UD 7311753 IC50 < 50000000 nM T70977 CY20RA 7458031 IC50 = 176 nM T70977 C2B4OG 7857292 IC50 = 65 nM T70977 CAY59K 8271528 IC50 > 10000 nM T70977 CG28IF 9599906 IC50 = 100 nM T70977 C1V4JH 9604909 IC50 = 75000 nM T70977 C36CFU 9604910 IC50 = 100000 nM T70977 CSP32E 9604911 IC50 = 6.31 nM T70977 C7G4PE 9604917 IC50 = 100 nM T70977 CT5QE7 9604918 IC50 = 158.49 nM T70977 C7Q8GN 9604919 IC50 = 158.49 nM T70977 CI8G9N 9604920 IC50 > 31622.78 nM T70977 CATL63 9604921 IC50 = 2511.89 nM T70977 CYFU08 9604922 IC50 = 7.943 nM T70977 CC3XQ1 9604923 IC50 = 1000 nM T70977 CMV30J 9604924 IC50 = 100 nM T70977 C6S2LW 9604925 IC50 = 316.23 nM T70977 CA4FS6 9604926 IC50 = 3981.07 nM T70977 CA58ZK 9604927 IC50 = 1995.26 nM T70977 C94LKU 9604928 IC50 = 158.49 nM T70977 CMN8A6 9604929 IC50 = 630.96 nM T70977 COP69S 9604930 IC50 = 316.23 nM T70977 CSV36K 9604931 IC50 = 251.19 nM T70977 CMD16A 9604932 IC50 > 31622.78 nM T70977 C6DUS1 9604933 IC50 = 1258.93 nM T70977 CQGN49 9604934 IC50 = 31.62 nM T70977 CPG6A5 9604935 IC50 = 3.162 nM T70977 CS83ME 9604936 IC50 = 39.81 nM T70977 C68ERA 9604937 IC50 = 39.81 nM T70977 CIW3B9 9604938 IC50 = 10 nM T70977 C10ZGV 9604939 IC50 > 25118.86 nM T70977 CWI97L 9604940 IC50 = 25.12 nM T70977 C24SBX 9604941 IC50 = 31.62 nM T70977 CX73WZ 9604942 IC50 = 125.89 nM T70977 CM53VP 9604943 IC50 = 7.943 nM T70977 CQT75V 9604944 IC50 = 15.85 nM T70977 C8P7UH 9604945 IC50 = 10 nM T70977 CP2M5R 9604946 IC50 = 2.512 nM T70977 CUR3T6 9604947 IC50 = 3.981 nM T70977 CTO5K7 9604948 IC50 = 2.512 nM T70977 CNS72D 9604949 IC50 = 158.49 nM T70977 CG6U7Z 9604950 IC50 = 2511.89 nM T70977 CAHN38 9604951 IC50 = 6.31 nM T70977 CI5DR9 9604952 IC50 = 2511.89 nM T70977 C2J4AK 9604953 IC50 = 5.012 nM T70977 COSU96 9604954 IC50 = 3.981 nM T70977 C4US0G 9604955 IC50 = 12.59 nM T70977 CQE07K 9604956 IC50 = 15.85 nM T70977 CJ1Q6P 9604957 IC50 = 5.012 nM T70977 C1YZ0I 9604958 IC50 > 31622.78 nM T70977 CB0H9G 9604959 IC50 > 31622.78 nM T70977 CX3TW8 9604960 IC50 = 15.85 nM T70977 CQ8N6O 9604961 IC50 = 31.62 nM T70977 C1CNW2 9604962 IC50 = 15.85 nM T70977 CH9O5R 9604963 IC50 = 7.943 nM T70977 CU17BF 9604964 IC50 = 10 nM T70977 CJM2X6 9604965 IC50 = 10 nM T70977 CW4TU6 9604966 IC50 = 12.59 nM T70977 CF7ZL3 9604967 IC50 = 10 nM T70977 C5ZS2I 9604968 IC50 = 31.62 nM T70977 C1R8QZ 9604969 IC50 = 63.1 nM T70977 CUO29M 9604970 IC50 = 6309.57 nM T70977 C6XK0Q 9795144 IC50 = 2400 nM T70977 CBT0X5 9797847 IC50 = 4380 nM T70977 CU7ZH6 9817982 IC50 = 90 nM T70977 C6Q2LF 9822667 IC50 = 36 nM T70977 C31XGW 9825189 IC50 = 460 nM T70977 C41QWA 9857146 IC50 = 2200 nM T70977 C30ILC 9858224 IC50 = 1900 nM T70977 C1QM0N 9858715 Ki = 312 nM T70977 COH4Z7 9869237 EC50 = 400 nM T70977 CM5Z8X 9869943 IC50 > 1000 nM T70977 CMS3F1 9880962 IC50 = 25 nM T70977 C0PT9E 9882994 IC50 = 70 nM T70977 C7AR9S 9889536 IC50 = 640 nM T70977 CUG5J1 9901007 Ki = 73 nM T70977 C7UIP5 9901505 Ki = 51 nM T70977 C2Y3WG 9907612 IC50 = 23000 nM T70977 CM5DB8 9909749 IC50 = 54 nM T70977 C61WVO 9923750 IC50 = 38 nM T70977 CA05BZ 9925230 Ki = 124 nM T70977 CSB0O2 9928879 IC50 = 70 nM T70977 CQD2W7 9935079 IC50 = 21.88 nM T70977 CS5KX9 9938299 IC50 > 10000 nM T70977 CDT67L 9947412 Ki = 33 nM T70977 CJO47T 9948405 IC50 > 10000 nM T70977 C75QCM 9969776 Ki = 605 nM T70977 CD29OS 9975371 IC50 = 31 nM T70977 CM5EI2 9976396 IC50 = 310 nM T70977 CJ84TX 9977154 IC50 = 10 nM T70977 C2W3AV 9995236 IC50 = 2500 nM T70977 CV8I5X 9999342 IC50 > 10000 nM T70977 CJ2EP9 9999648 EC50 = 390 nM T70977 C5XU8E 10000872 IC50 = 31 nM T70977 C57DLH 10001523 IC50 = 15 nM T70977 C84CYF 10001880 IC50 = 14 nM T70977 CBT2P7 10001889 IC50 = 65 nM T70977 CV7Z9Y 10002471 IC50 = 140 nM T70977 CCL6W3 10006844 Ki = 690 nM T70977 C4A5SD 10040883 IC50 > 100000 nM T70977 C4VXU1 10041379 IC50 = 2700 nM T70977 C3U7AR 10043221 IC50 = 420 nM T70977 CTSH96 10044516 IC50 = 2000 nM T70977 C9XG7U 10052336 Ki = 12 nM T70977 CO5KL3 10072710 IC50 = 20 nM T70977 CINF40 10073694 IC50 = 7 nM T70977 CTHZ45 10087157 IC50 = 55000 nM T70977 CPB50A 10110392 IC50 = 2200 nM T70977 CZV3U5 10111694 Ki = 113 nM T70977 CV9B4X 10112611 Ki = 338 nM T70977 CNK72I 10113102 Ki = 4.4 nM T70977 CFXZ38 10114332 IC50 = 620 nM T70977 CEF8U5 10117705 IC50 = 71 nM T70977 CGUV49 10118014 Ki = 0.46 nM T70977 CIF96U 10118131 Ki = 8.4 nM T70977 CR6EP2 10118731 Ki = 1.5 nM T70977 CRT67V 10119173 IC50 = 40 nM T70977 CF9A5O 10125353 Ki = 690 nM T70977 CO6E1A 10125856 IC50 = 25000 nM T70977 C0H9JX 10125875 IC50 = 10000 nM T70977 CTXW95 10126509 IC50 = 200 nM T70977 CB4Y3W 10131935 IC50 = 52 nM T70977 CRW07C 10133485 IC50 = 27 nM T70977 CLA2N6 10133600 Ki = 44 nM T70977 CKL3V4 10134576 Ki > 150 nM T70977 CM49JT 10138033 Ki = 0.4 nM T70977 CI4SG5 10139085 Ki = 18 nM T70977 CKUD10 10139154 Ki = 16 nM T70977 CZJI60 10141037 IC50 = 34 nM T70977 CW3MD1 10141178 Ki = 74 nM T70977 C42TSU 10142642 Ki = 0.48 nM T70977 C94WRY 10143231 IC50 = 34 nM T70977 C76TVG 10143584 IC50 = 890 nM T70977 CY7W1Z 10144680 IC50 = 51 nM T70977 CLBD08 10144909 IC50 = 2400 nM T70977 CM79VS 10149184 Ki > 3300 nM T70977 CV73FD 10157920 Ki > 15 nM T70977 C69DHW 10158652 IC50 < 16000 nM T70977 CQN8M3 10159519 Ki = 67 nM T70977 C7JP1A 10163439 IC50 = 150 nM T70977 CTIP10 10164394 Ki = 1.3 nM T70977 CC8XJ5 10171595 Ki = 620 nM T70977 CB28QI 10171783 Ki > 3300 nM T70977 CL7FI4 10171832 Ki > 5000 nM T70977 CQG5R4 10173796 IC50 = 16 nM T70977 CO4AS3 10177172 Ki = 12 nM T70977 CQ6J1C 10179215 Ki = 48 nM T70977 C3KHT0 10179373 Ki = 1500 nM T70977 CXD4Z2 10180161 Ki = 1314 nM T70977 CO08KZ 10182284 Ki > 4000 nM T70977 CB8MU3 10182620 Ki = 3.1 nM T70977 C3QZV8 10184859 IC50 = 270 nM T70977 CJN72C 10185160 IC50 = 370 nM T70977 CJ0R2G 10187378 IC50 = 4800 nM T70977 C73LXY 10188021 IC50 = 2500 nM T70977 CK7UT9 10188786 IC50 = 1200 nM T70977 CY7W5M 10192938 IC50 = 3200 nM T70977 CYG69U 10193464 IC50 = 25000 nM T70977 CHP56L 10193482 IC50 = 32000 nM T70977 C7PEG0 10200408 Ki = 1034 nM T70977 C5P8JC 10206423 IC50 = 16.98 nM T70977 C63OAC 10207408 Ki = 6.3 nM T70977 CGOT91 10207821 IC50 = 25 nM T70977 CUF0W9 10207822 IC50 = 4 nM T70977 C0IYO3 10208648 IC50 = 26 nM T70977 C51SKM 10209082 IC50 = 1900 nM T70977 CK72XG 10209108 IC50 = 1300 nM T70977 CBJ87W 10214957 IC50 = 1000 nM T70977 C51UXK 10215135 IC50 = 25000 nM T70977 COWF65 10215271 IC50 = 2 nM T70977 CIHO38 10215426 IC50 = 5000 nM T70977 C1Z6EJ 10222721 Ki = 8 nM T70977 C3VK7T 10229967 IC50 = 43 nM T70977 CX8YO7 10231705 Ki = 0.22 nM T70977 CJ39UQ 10236371 Ki = 240 nM T70977 C1LB5O 10236721 IC50 = 3000 nM T70977 C6NV7Q 10236923 IC50 > 32000 nM T70977 CTS43G 10238877 IC50 > 25000 nM T70977 CH48JA 10239038 IC50 = 690 nM T70977 CK4N5M 10247132 IC50 = 480 nM T70977 C5TQ7X 10247543 IC50 > 10000 nM T70977 C8PJ1V 10248119 IC50 = 270 nM T70977 C9HJ3N 10248940 IC50 = 37 nM T70977 CD6WK8 10249180 IC50 = 570 nM T70977 CY27WR 10250197 IC50 = 1160 nM T70977 C6J9YK 10254786 Ki = 22 nM T70977 C3LY6S 10256075 IC50 = 80 nM T70977 CCO9Y4 10263500 IC50 = 6800 nM T70977 CRUF54 10264733 IC50 = 7010 nM T70977 CGF6I3 10267834 Ki = 24 nM T70977 C28AEC 10268530 Ki = 171 nM T70977 CLQ3P2 10270356 Ki = 126 nM T70977 CC7P0T 10272623 IC50 = 200 nM T70977 C2X6LY 10275064 IC50 = 136 nM T70977 C14JRY 10275824 Ki = 64 nM T70977 C7U9BE 10281603 IC50 = 403 nM T70977 C8GJ9A 10286242 IC50 > 32000 nM T70977 C42MKP 10286399 IC50 = 25000 nM T70977 C2O4LF 10286648 IC50 > 32000 nM T70977 CF9N7Y 10292186 Ki = 216 nM T70977 C7SFI1 10296883 IC50 = 870 nM T70977 CTXN56 10296960 IC50 = 49 nM T70977 C45WIV 10297008 Ki = 0.67 nM T70977 C4F1YI 10297128 IC50 = 138 nM T70977 CIB8P4 10301015 Ki = 9 nM T70977 C8RD3V 10301884 IC50 > 10000 nM T70977 CAX9W2 10302405 IC50 = 3900 nM T70977 C9RK8E 10303030 Ki = 1.1 nM T70977 CZS4V6 10308171 IC50 = 25000 nM T70977 C9MVA5 10308281 IC50 = 25000 nM T70977 CKA8B0 10308522 IC50 = 10 nM T70977 CD3ER5 10308589 IC50 = 8.9 nM T70977 COD9W2 10308706 IC50 = 50 nM T70977 C9GP1M 10309005 IC50 = 13 nM T70977 CH0I3K 10309738 IC50 = 2000 nM T70977 C6S9AO 10310395 IC50 = 850 nM T70977 CNE1H0 10318765 IC50 = 6 nM T70977 C3IJR7 10339551 IC50 = 4 nM T70977 CHB84X 10341165 IC50 = 8 nM T70977 CD5G7Z 10355643 IC50 = 1180 nM T70977 C5GTM6 10366534 IC50 = 26 nM T70977 CO4UF0 10367481 Ki = 90 nM T70977 CWUM08 10380356 IC50 = 500 nM T70977 CYB64W 10382823 IC50 = 870 nM T70977 CSK76I 10403564 IC50 = 3530 nM T70977 CRVE78 10411641 IC50 = 14 nM T70977 CYIV48 10412503 IC50 = 6000 nM T70977 C2B0IU 10421236 IC50 = 1300 nM T70977 C7HBP6 10429593 IC50 = 3630 nM T70977 CW5SJ3 10430664 IC50 = 280 nM T70977 C6I8SW 10435170 IC50 = 450 nM T70977 C1V9GY 10446453 IC50 > 10000 nM T70977 CITG13 10452673 IC50 = 1184 nM T70977 CYJ49W 10459291 Ki = 74 nM T70977 C0N3UL 10471927 IC50 = 920 nM T70977 C2WQ8M 10473563 IC50 > 10000 nM T70977 CV9ZL0 10475216 IC50 = 480 nM T70977 C9BHN2 10533009 IC50 = 530 nM T70977 C47NIR 10801110 IC50 = 1100 nM T70977 CJ3Q6V 10862509 IC50 > 250000 nM T70977 CE3UD1 10894181 IC50 = 240 nM T70977 C96WQF 10894235 IC50 = 100 nM T70977 CHW8D4 10902866 IC50 = 50000 nM T70977 CDO1N6 10904317 IC50 = 6920 nM T70977 CK83OD 10904406 IC50 = 15 nM T70977 CWH1Q8 10948459 IC50 = 1000 nM T70977 C94ANH 10965763 IC50 = 420000 nM T70977 C5HG2R 11101023 IC50 = 2100 nM T70977 CWUN25 11152016 Ki = 16000 nM T70977 C94QUD 11163861 Ki = 10 nM T70977 CHJP46 11164978 IC50 = 1.1 nM T70977 CJEW09 11176034 IC50 = 22 nM T70977 CAG98O 11187702 IC50 = 8.6 nM T70977 C04NLR 11245667 IC50 > 50000 nM T70977 C30PKR 11248978 IC50 = 2.6 nM T70977 CRU8F6 11269073 IC50 = 1.7 nM T70977 CMZ6Q7 11277469 IC50 = 11000 nM T70977 C6C3JX 11281930 IC50 > 10000 nM T70977 CJP4C1 11283328 IC50 = 0.3 nM T70977 CHB2U6 11284129 IC50 = 5300 nM T70977 CSXY78 11294864 IC50 = 1.6 nM T70977 C81TUN 11303752 IC50 = 410 nM T70977 C1X5OV 11315047 IC50 = 6.6 nM T70977 CJXV31 11315049 IC50 = 9.6 nM T70977 CPU9I3 11316975 IC50 = 12 nM T70977 CN4TU7 11328055 IC50 = 1700 nM T70977 CQ8I4H 11328863 IC50 = 1.3 nM T70977 C19GSN 11349589 IC50 = 2.6 nM T70977 CUM15V 11358339 IC50 > 50000 nM T70977 CE8VP2 11361885 IC50 = 300 nM T70977 C43NPS 11373886 IC50 > 10000 nM T70977 C8KPE4 11380176 IC50 > 50000 nM T70977 CJ3O0G 11384249 IC50 = 5.2 nM T70977 CG1T5J 11386640 IC50 = 3400 nM T70977 CVI1A3 11395082 IC50 = 180 nM T70977 CFOZ52 11407074 IC50 = 50 nM T70977 CE7QB2 11429096 IC50 = 27 nM T70977 C4PSB5 11437879 IC50 > 50000 nM T70977 CVN1C0 11477611 IC50 = 4000 nM T70977 C6K0GD 11484301 IC50 = 2800 nM T70977 CJNM24 11485846 IC50 = 5.4 nM T70977 CXT91K 11488074 IC50 = 50000 nM T70977 CS2YO1 11492918 Ki > 3300 nM T70977 C0H6QS 11495680 IC50 > 10000 nM T70977 CIW9L5 11502867 IC50 > 10000 nM T70977 CK2Q0X 11516978 IC50 > 10000 nM T70977 CPE53F 11526238 IC50 > 10000 nM T70977 CL7X4Q 11530963 IC50 = 71 nM T70977 C5BM4T 11531799 IC50 > 10000 nM T70977 C53OSD 11532048 IC50 > 10000 nM T70977 CC4QM5 11532676 IC50 > 10000 nM T70977 CCJ7Z1 11535873 IC50 > 30000 nM T70977 CTG83F 11539329 Ki > 7100 nM T70977 C01FVM 11546457 IC50 > 10000 nM T70977 C6FJU5 11560568 IC50 = 0.6 nM T70977 CACS26 11561968 Ki = 1900 nM T70977 CNBM81 11562171 IC50 > 10000 nM T70977 C3WVM7 11564772 IC50 = 15000 nM T70977 C4LI8C 11564882 IC50 = 11000 nM T70977 CD3E8M 11574606 IC50 = 190 nM T70977 CMIL86 11590363 Ki > 7100 nM T70977 C0NV9Y 11596881 IC50 > 10000 nM T70977 CU7WH8 11601694 IC50 = 628 nM T70977 C71WAD 11615485 Ki = 690 nM T70977 C93UKS 11617172 IC50 = 200 nM T70977 C1BLZ5 11620055 IC50 > 10000 nM T70977 C5B3XJ 11620410 IC50 > 40000 nM T70977 C9T6SC 11640926 Ki > 7100 nM T70977 C24GRQ 11661959 IC50 > 10000 nM T70977 CAS3D2 11666764 IC50 = 3000 nM T70977 CC5B1E 11681688 IC50 = 1300 nM T70977 CS72ED 11682843 IC50 > 10000 nM T70977 CU0E8O 11690457 Ki = 400 nM T70977 CLC53E 11691173 IC50 > 10000 nM T70977 C65FVB 11694317 Ki > 3300 nM T70977 CPK2W8 11696113 IC50 = 1400 nM T70977 CB0AP2 11705863 Ki = 2100 nM T70977 CM49IK 11715597 IC50 > 30000 nM T70977 C9UA2S 11718220 IC50 = 280 nM T70977 C1FTX3 11719305 IC50 > 10000 nM T70977 C0ZJD8 11731783 IC50 = 11700 nM T70977 C3I2RM 11747156 IC50 > 100000 nM T70977 CU1O9G 11748865 IC50 = 18 nM T70977 CP7AH3 11755812 IC50 = 50000 nM T70977 C1FUP2 11760761 IC50 = 9300 nM T70977 CL81HQ 11819216 IC50 = 700 nM T70977 C9VRK1 11822355 IC50 > 1000000 nM T70977 C9JT4S 11847343 IC50 > 10000 nM T70977 CTI2R7 11856271 IC50 = 198 nM T70977 C64JCR 11856273 IC50 = 41 nM T70977 COT84C 11856529 IC50 = 125 nM T70977 CD9A7C 11856530 IC50 = 230 nM T70977 C9A6KM 11857236 IC50 = 80 nM T70977 CA9ST2 11959186 IC50 = 1210 nM T70977 CC7M0D 11959190 IC50 = 400 nM T70977 C39VTW 11959283 IC50 = 1020 nM T70977 CQ8U1P 11959284 IC50 = 303 nM T70977 C36HDX 11959286 IC50 = 13200 nM T70977 CTE96C 11959310 IC50 = 4000 nM T70977 CO0A4K 11959314 IC50 = 40 nM T70977 C12CRJ 11959377 IC50 = 2700 nM T70977 CUWL12 11959378 IC50 = 375 nM T70977 CVPT94 11959513 IC50 = 30000 nM T70977 C5LZ9C 11959550 IC50 = 30000 nM T70977 C3UVQ2 11959600 IC50 = 2600 nM T70977 C1WDQ0 11959682 IC50 = 1040 nM T70977 CMW89V 11959683 IC50 = 1110 nM T70977 CA6K4Y 11959684 IC50 = 310 nM T70977 CW53JC 11998038 Ki = 210 nM T70977 CK0GN2 12018144 IC50 = 1 nM T70977 C4H7YC 12018155 IC50 = 0.4 nM T70977 CM7FP9 12128595 IC50 > 50000 nM T70977 C82APV 12373568 IC50 = 75000 nM T70977 C2MCR0 12374705 IC50 = 12750 nM T70977 CP62DO 12616884 IC50 = 980 nM T70977 C0W9EM 12629212 IC50 > 100000 nM T70977 CSU6V2 12807269 IC50 = 138 nM T70977 CFMC48 12867665 IC50 > 100000 nM T70977 CTC7D9 13091616 IC50 > 100000 nM T70977 CHJ01P 13303387 IC50 > 10000 nM T70977 C5YF0D 13303393 IC50 > 10000 nM T70977 CQ0Z5X 13901969 IC50 > 1000 nM T70977 C0L9RB 13954062 IC50 = 12940 nM T70977 CE86GH 14951779 IC50 = 1378 nM T70977 C6JIA9 14977359 IC50 = 24360 nM T70977 C23IYJ 15314149 IC50 > 10000 nM T70977 CH0M1O 15604545 IC50 > 100000 nM T70977 C58VZQ 15604546 IC50 > 100000 nM T70977 CV0DW1 15948777 IC50 > 1000 nM T70977 C7LB4I 15949613 IC50 > 10000 nM T70977 CFPW41 16007116 Ki > 7000 nM T70977 CWR60H 16010405 IC50 > 100000 nM T70977 C9TU1O 16046126 IC50 = 13 nM T70977 C5VPH9 16129448 IC50 = 9410 nM T70977 C9FMS4 16374676 IC50 = 3162 nM T70977 C5S6BM 16664484 IC50 >= 12400 nM T70977 CU56EW 16664858 IC50 > 10000 nM T70977 CC24KI 16667248 IC50 = 6 nM T70977 CC8S9V 16734945 IC50 = 3 nM T70977 CG95IN 16738711 IC50 = 45 nM T70977 CI3F1J 16741475 IC50 = 7 nM T70977 C0K5HJ 16741476 IC50 = 15 nM T70977 C5UY9I 16741552 IC50 = 42 nM T70977 CYQ9W5 16741728 IC50 = 235 nM T70977 C9KNO4 16741730 IC50 = 55 nM T70977 C3OP0J 16751208 IC50 = 10690 nM T70977 C9IK2X 16758212 IC50 = 15 nM T70977 CB7U1R 17408143 IC50 = 521 nM T70977 C1W0AL 17592753 IC50 > 50000 nM T70977 C9C5TV 17751819 IC50 = 660 nM T70977 CWH37T 17758574 IC50 > 10000 nM T70977 CM3BG9 18521798 IC50 = 1000 nM T70977 C47YSL 18669003 IC50 = 6130 nM T70977 CFA8M9 18768052 IC50 = 3200 nM T70977 C7CLY0 18780230 IC50 = 42 nM T70977 CVT26W 19167508 IC50 = 7080 nM T70977 C3YER4 19696390 IC50 = 10 nM T70977 C0CGB9 20878104 IC50 > 100000 nM T70977 CSE90B 20878299 IC50 = 77200 nM T70977 CN29WK 20963524 IC50 = 1000 nM T70977 C6ER5O 21065569 IC50 = 500 nM T70977 CD76CS 21065645 IC50 = 1100 nM T70977 C41LUC 21066960 IC50 = 247 nM T70977 CUDH82 21067035 IC50 = 1130 nM T70977 C40VQC 21067040 IC50 = 1410 nM T70977 CJ17WY 21067041 IC50 = 1180 nM T70977 CP97QM 21067220 IC50 = 4600 nM T70977 C7XJ8M 21067235 IC50 = 9820 nM T70977 C06VOI 21067290 IC50 = 790 nM T70977 CL81VC 21100709 IC50 = 2630 nM T70977 CC2UB6 21214332 IC50 = 1193 nM T70977 CY6CQ1 21214334 IC50 = 405 nM T70977 C8IF5U 21991073 Ki = 1168 nM T70977 C5NFB1 22319486 IC50 = 3808 nM T70977 C5JS0Q 22319495 IC50 = 12247 nM T70977 C2REA5 22319512 IC50 = 1720000 nM T70977 CYT10Z 22319523 IC50 = 10546 nM T70977 CQ1I9E 22319541 IC50 = 18000 nM T70977 CV92RI 22319550 IC50 = 23000 nM T70977 C78SRF 22319555 IC50 = 5498 nM T70977 C3UP4L 22319556 IC50 > 100000 nM T70977 C62SME 22319558 IC50 > 100000 nM T70977 CB5OK1 22319566 IC50 = 7165 nM T70977 CQ9S6R 22319587 IC50 > 100000 nM T70977 CR68LU 22319598 IC50 = 12000 nM T70977 CR1J3V 22319606 IC50 = 16784 nM T70977 CFUD85 22319607 IC50 = 80 nM T70977 CQ5G2Y 22319619 IC50 = 1088 nM T70977 C70MVP 22319622 IC50 = 30 nM T70977 C9KDP8 22319661 IC50 = 8000 nM T70977 CKL69A 22319674 IC50 = 130 nM T70977 C6HZ0M 22319680 IC50 = 50000 nM T70977 C49VCU 22319691 IC50 = 5413 nM T70977 C3AE1U 22521053 IC50 = 5000 nM T70977 CJ52OX 22521086 IC50 = 2000 nM T70977 C2KEA7 22521089 IC50 = 710 nM T70977 C6Z9SJ 22595645 IC50 = 23 nM T70977 CDSV36 22595656 IC50 = 150 nM T70977 C6XHE4 22595681 IC50 = 39 nM T70977 CG3KB2 22595683 IC50 = 130 nM T70977 CUS76C 22607543 IC50 > 10000 nM T70977 COW84Q 22712543 IC50 = 1000 nM T70977 C42OBN 23586145 IC50 = 29000 nM T70977 CN39TP 23586146 IC50 = 970 nM T70977 C28MIO 23643730 IC50 = 8500 nM T70977 CGC1I7 23645297 IC50 > 100000 nM T70977 CSTI83 23645298 IC50 > 100000 nM T70977 CC3V0P 23645299 IC50 > 100000 nM T70977 CIA9Q3 23645300 IC50 > 100000 nM T70977 C7XJ4I 23645301 IC50 > 100000 nM T70977 C9R4WS 23645302 IC50 > 100000 nM T70977 C5WC7V 23645303 IC50 > 100000 nM T70977 CL2T3I 23645566 IC50 = 22000 nM T70977 C16MYH 23645567 IC50 = 5100 nM T70977 CV3Q1Z 23645568 IC50 > 50000 nM T70977 CR53PW 23645569 IC50 > 50000 nM T70977 CM20NA 23645570 IC50 = 28000 nM T70977 CMJ4C7 23645571 IC50 > 50000 nM T70977 CBK47A 23645572 IC50 = 50000 nM T70977 CR5I7U 23645573 IC50 = 12000 nM T70977 CE7QN6 23645574 IC50 = 8700 nM T70977 C6YF5D 23645577 IC50 = 11000 nM T70977 C9G5EQ 23645578 IC50 = 780 nM T70977 C95CXB 23645579 IC50 = 20000 nM T70977 CHK57M 23645580 IC50 = 43000 nM T70977 CG6D4M 23647319 IC50 > 10000 nM T70977 CY8Z7X 23647330 IC50 > 10000 nM T70977 C4XD8H 23647348 IC50 > 10000 nM T70977 C2WU3S 23729136 IC50 = 3.1 nM T70977 C25DMJ 24180565 IC50 = 25 nM T70977 CFMQ08 24370907 IC50 = 83 nM T70977 CZKX63 24746470 IC50 = 30 nM T70977 CKW2O0 24746471 IC50 = 11 nM T70977 C61QMV 24746472 IC50 = 24 nM T70977 C04GKS 24746625 IC50 = 37 nM T70977 C8QD5W 24746626 IC50 = 7 nM T70977 CZ6G2H 24748456 Ki = 370 nM T70977 C52FSU 24752942 IC50 = 270 nM T70977 CR8A5O 24752945 IC50 = 1000 nM T70977 C0YX4T 24752946 IC50 = 13 nM T70977 CD10JY 24753107 IC50 = 440 nM T70977 CHRF96 24753108 IC50 = 900 nM T70977 C36RZG 24753109 IC50 = 100 nM T70977 C7S2VU 24753198 IC50 = 190 nM T70977 C6F1LP 24753200 IC50 = 600 nM T70977 CVZ7Q5 24753289 IC50 = 660 nM T70977 CJIV04 24753375 IC50 = 110 nM T70977 C9BE6G 24753378 IC50 = 290 nM T70977 CC05GK 24753463 IC50 = 45 nM T70977 CIZ98W 24753666 IC50 = 47 nM T70977 CA3I4T 24753787 IC50 > 50000 nM T70977 CIJ9A5 24753849 IC50 = 22 nM T70977 CVTK64 24754021 IC50 = 65 nM T70977 CNYI28 24754024 IC50 = 31 nM T70977 C5S9FI 24754025 IC50 = 160 nM T70977 C7YG1N 24759534 IC50 = 220 nM T70977 C7R9TA 24762195 IC50 = 500 nM T70977 C0VZQ5 24765998 IC50 = 227 nM T70977 CPJB16 24768116 IC50 > 5000 nM T70977 CH58ID 24768117 IC50 > 5000 nM T70977 C1ZJT0 24768118 IC50 > 5000 nM T70977 CKJ8O1 24768119 IC50 > 5000 nM T70977 CR7VX5 24768120 IC50 > 2000 nM T70977 C7WA9T 24768121 IC50 > 5000 nM T70977 CA52ER 24768122 IC50 > 5000 nM T70977 CS7CV8 24782785 EC50 = 50 nM T70977 C7QWR2 24783299 EC50 = 290 nM T70977 CZG70Y 24784075 EC50 = 31 nM T70977 CBC6A1 24784328 EC50 = 150 nM T70977 C2O3WZ 24784332 IC50 = 44 nM T70977 CP8Y0H 24784579 IC50 = 27 nM T70977 CLBP72 24798571 IC50 = 7114 nM T70977 C9QMJ6 24809762 IC50 < 100 nM T70977 CI5B6S 24825779 IC50 = 247 nM T70977 C1H2AM 24828716 IC50 > 30000 nM T70977 CU9E4W 24828717 IC50 = 590 nM T70977 C5U2ZM 24828854 IC50 = 1700 nM T70977 C57SYK 24829098 IC50 = 7500 nM T70977 CM5AX9 24829102 IC50 = 1400 nM T70977 CY97JK 24829220 IC50 < 1000 nM T70977 C5IA6Q 24851353 IC50 = 3.981 nM T70977 CCGY62 24860825 IC50 = 1050 nM T70977 CC9V2Y 24882562 IC50 = 920 nM T70977 CY8L7E 24896769 IC50 > 10000 nM T70977 C7N4DI 24959043 IC50 > 100000 nM T70977 C6CVK4 24959046 IC50 > 100000 nM T70977 CV5IE4 24963049 IC50 = 41 nM T70977 CVI75F 24991569 IC50 = 3.5 nM T70977 CAC94U 24991573 IC50 = 34.5 nM T70977 C0NAG9 24991913 IC50 = 16.1 nM T70977 CGM47T 24991914 IC50 = 440 nM T70977 CRK3U5 24991915 IC50 = 223 nM T70977 C4FUW2 24991916 IC50 = 830 nM T70977 C4EG8R 24993189 IC50 > 10000 nM T70977 CJ1ZU3 25004596 IC50 = 13 nM T70977 CP0Q8F 25004597 IC50 = 29 nM T70977 C3SB8A 25004925 IC50 = 80 nM T70977 C4PKF3 25004926 IC50 = 920 nM T70977 CL7P6C 25004927 IC50 = 76 nM T70977 C3EZ5A 25004929 IC50 = 22 nM T70977 C53GVH 25004931 IC50 > 1000 nM T70977 C3DMZ4 25005268 IC50 > 1000 nM T70977 C2BPD5 25005270 IC50 = 21 nM T70977 C5PC0U 25005271 IC50 = 49 nM T70977 CNYP16 25005272 IC50 = 46 nM T70977 CT64BR 25005273 IC50 = 19 nM T70977 CZOS89 25005627 IC50 = 70 nM T70977 CX0O4A 25005628 IC50 = 8.3 nM T70977 CR9LQ8 25005629 IC50 = 1.4 nM T70977 CWBO80 25005631 IC50 = 0.2 nM T70977 C8ZQ3E 25005985 IC50 = 0.5 nM T70977 C47CFM 25005986 IC50 = 0.4 nM T70977 CKT5V7 25005987 IC50 = 0.8 nM T70977 C5NF9P 25005988 IC50 = 0.2 nM T70977 C2H8XF 25005989 IC50 = 0.1 nM T70977 C1MWK0 25005990 IC50 = 13 nM T70977 CQ1OY4 25006369 IC50 = 780 nM T70977 CY8RC1 25022535 IC50 = 23 nM T70977 CM57PT 25032775 IC50 = 2200 nM T70977 CTV54O 25123227 IC50 > 10000 nM T70977 C78YWA 25145716 IC50 > 500 nM T70977 CB21XV 25164469 Ki = 265 nM T70977 CNF0A8 25164674 Ki = 4272 nM T70977 CUX83H 25164675 Ki = 572 nM T70977 C1H7BF 25164677 Ki = 2530 nM T70977 CN50EI 25164678 Ki = 3402 nM T70977 C3XI7P 25164880 Ki > 5450 nM T70977 CX80QK 25164883 Ki = 10 nM T70977 C6SD2A 25165081 Ki = 3810 nM T70977 C67TVH 25165085 Ki = 542 nM T70977 C8J4KL 25165278 Ki = 450 nM T70977 CRJ6M7 25165279 Ki > 5450 nM T70977 C7RBX0 25165280 Ki > 5450 nM T70977 CPEY29 25165481 Ki > 5450 nM T70977 C70DRX 25165482 Ki > 5450 nM T70977 CE8D1W 25165860 Ki = 448 nM T70977 C6VZU2 25165861 Ki = 39 nM T70977 CVI70X 25166053 Ki = 70 nM T70977 C9VA1N 25166056 Ki = 91 nM T70977 C1JS9O 25166057 Ki = 26 nM T70977 CM41PX 25166058 Ki = 70 nM T70977 CT94MS 25166059 Ki = 45 nM T70977 C5BM7F 25166250 Ki = 23 nM T70977 CCN25J 25166251 Ki = 197 nM T70977 CX8HY9 25166657 Ki = 48 nM T70977 C1CNX7 25166659 Ki = 16 nM T70977 C81WIV 25166867 Ki = 28 nM T70977 C9MR2O 25166869 Ki = 642 nM T70977 CAG1H6 25166870 Ki = 2611 nM T70977 CGUC69 25167072 Ki = 10 nM T70977 CF4G1L 25167074 Ki = 17 nM T70977 C35ZXL 25167075 Ki = 289 nM T70977 C1CRJ7 25167076 Ki = 2861 nM T70977 C1IFX5 25167077 Ki = 3925 nM T70977 C2D3FP 25167078 Ki > 5450 nM T70977 CP2W8I 25167079 Ki = 4472 nM T70977 CJO5A4 25167275 Ki > 5450 nM T70977 C5KX0G 25167277 Ki = 19 nM T70977 CQ5FJ8 25167278 Ki = 121 nM T70977 C37YSX 25167280 Ki = 141 nM T70977 C0OW7X 25167905 IC50 = 3 nM T70977 CY9ZF2 25169385 IC50 = 350 nM T70977 C4ZQ9E 25169520 IC50 = 410 nM T70977 C0X3KV 25181321 IC50 = 2.3 nM T70977 CHN5O0 25190977 IC50 = 560 nM T70977 CD4J7S 25195477 EC50 = 20000 nM T70977 CT3XE1 25199517 IC50 > 100000 nM T70977 C6FGQ1 25206346 IC50 > 10000 nM T70977 CNG96H 25210579 IC50 > 10000 nM T70977 CVNK24 25210880 IC50 = 310 nM T70977 C0GL7R 25212179 IC50 = 548 nM T70977 C87NZS 25212180 IC50 = 467 nM T70977 C9A3ED 25216880 IC50 > 50000 nM T70977 COWB90 25221040 IC50 = 280 nM T70977 CC25TV 25222706 IC50 = 680 nM T70977 CH9IB2 25253663 IC50 = 57 nM T70977 C1WQ7R 25253819 IC50 = 37 nM T70977 CJ7UH1 25253821 IC50 = 250 nM T70977 C4D0OG 25253822 EC50 = 1400 nM T70977 C2Q9YM 25253823 EC50 = 2100 nM T70977 C42JQD 25253980 IC50 = 550 nM T70977 C7VG2M 25264966 IC50 = 20 nM T70977 C3QWS0 25264968 IC50 = 2.4 nM T70977 CD6Y0G 25268197 IC50 > 50000 nM T70977 CR59TN 25268198 IC50 > 50000 nM T70977 C1DR5Z 25268199 IC50 > 50000 nM T70977 CV4N5C 25268555 IC50 > 50000 nM T70977 CPM85N 25268556 IC50 > 50000 nM T70977 CT7EB2 25268557 IC50 > 50000 nM T70977 CWB2K9 25268558 IC50 > 50000 nM T70977 C81HUL 25268559 IC50 > 50000 nM T70977 CC71QJ 27666048 IC50 > 100000 nM T70977 C2U0NP 30291209 IC50 = 39 nM T70977 C7S6OT 30291292 IC50 = 41 nM T70977 CU2B4F 42611245 IC50 >= 10000 nM T70977 CWS37O 42618140 IC50 > 25118.86 nM T70977 C2JV3O 42618143 IC50 > 25118.86 nM T70977 CG01BO 42618144 IC50 > 25118.86 nM T70977 CU9E4P 42629114 IC50 = 2.3 nM T70977 CO4FV0 42630578 IC50 > 25118.86 nM T70977 CGIT89 42630692 IC50 > 10000 nM T70977 CW0BO2 42630693 IC50 > 10000 nM T70977 CH93PI 43801944 IC50 > 10000 nM T70977 CO42DC 44138048 IC50 > 10000 nM T70977 CL65QV 44138049 IC50 > 10000 nM T70977 CB0O2A 44186880 Ki = 5216 nM T70977 C9K7OP 44186882 Ki = 2026 nM T70977 CX0ZU8 44186885 Ki = 3466 nM T70977 CNGV37 44189584 Ki > 5450 nM T70977 C8KNA3 44219632 Ki = 2900 nM T70977 C0VIX4 44219633 Ki = 230 nM T70977 C7TB2K 44219658 IC50 = 0.14 nM T70977 CEL61X 44229839 IC50 > 10000 nM T70977 CYE36B 44241613 IC50 = 140 nM T70977 C6LG5T 44241614 IC50 = 760 nM T70977 C7TX1L 44252656 Ki = 259 nM T70977 CIL1H2 44252657 IC50 = 92 nM T70977 CTP0E1 44307734 IC50 = 1.585 nM T70977 CLPC42 44334296 IC50 = 8 nM T70977 CF61IT 44334334 IC50 = 33 nM T70977 C50EFS 44334355 IC50 = 110 nM T70977 CH9SF8 44334367 IC50 = 31 nM T70977 C3BFI4 44334443 IC50 = 4 nM T70977 C4XG8M 44341125 IC50 > 250000 nM T70977 CEKJ39 44345742 IC50 = 3999.45 nM T70977 C0E9CV 44345921 IC50 = 500.03 nM T70977 CN2T9J 44345927 IC50 = 74.99 nM T70977 CV4D0J 44346042 IC50 = 41020.41 nM T70977 CSV1D5 44346075 IC50 = 349945.17 nM T70977 CQ2PI7 44346184 IC50 = 199.99 nM T70977 CCYJ71 44389363 IC50 = 5 nM T70977 CTS28N 44389373 IC50 = 11 nM T70977 CN0K1F 44389381 IC50 = 7.7 nM T70977 COG36F 44389387 IC50 = 0.7943 nM T70977 C0KN6M 44389389 IC50 = 297 nM T70977 C17KHC 44389424 IC50 = 38 nM T70977 C0TGU3 44389439 IC50 = 8.7 nM T70977 C7HTC6 44389448 IC50 = 4.2 nM T70977 C1MFZ6 44389453 IC50 = 111 nM T70977 C18ANZ 44389457 IC50 = 53 nM T70977 CSBC59 44396134 IC50 = 5.2 nM T70977 CV09DY 44410717 IC50 > 10000 nM T70977 CP3CI1 44410720 IC50 > 10000 nM T70977 C8W7AD 44410723 IC50 > 10000 nM T70977 CAT5X4 44410829 IC50 > 10000 nM T70977 CC6Y5P 44410844 IC50 > 10000 nM T70977 CG34TY 44410851 IC50 > 10000 nM T70977 C41EIA 44410869 IC50 > 10000 nM T70977 CB6AE8 44410948 IC50 > 10000 nM T70977 CXZG12 44410949 IC50 > 10000 nM T70977 CS7IE9 44410953 IC50 > 10000 nM T70977 CA9M4X 44410954 IC50 > 10000 nM T70977 C3SP5H 44410955 IC50 > 10000 nM T70977 C5D6YP 44410956 IC50 > 10000 nM T70977 C5W1VC 44410959 IC50 > 10000 nM T70977 CM1C2G 44410960 IC50 > 10000 nM T70977 CVSI80 44411048 IC50 > 10000 nM T70977 CN72BR 44411161 IC50 > 10000 nM T70977 C4AW0O 44411183 IC50 > 10000 nM T70977 COPG94 44427519 IC50 > 10000 nM T70977 C2HQ4O 44441925 IC50 = 580 nM T70977 CFX2T7 44441935 IC50 = 1000 nM T70977 C5OS1N 44444340 IC50 = 1800 nM T70977 C0I7AX 44444347 IC50 = 34 nM T70977 CZF15O 44444382 IC50 = 13310 nM T70977 CZJ8W0 44444384 IC50 = 15200 nM T70977 C5H9EK 44444385 IC50 = 35 nM T70977 CL4E9B 44444387 IC50 = 130 nM T70977 CG81QO 44444388 IC50 = 600 nM T70977 CN8J9C 44445395 IC50 = 16600 nM T70977 C5TR3Z 44445401 IC50 = 25000 nM T70977 CWD42G 44445991 IC50 = 320 nM T70977 CJ64MI 44445992 IC50 = 140 nM T70977 CS2G7K 44448292 IC50 = 13 nM T70977 C4E5DN 44448294 IC50 = 7 nM T70977 CU06RO 44448295 IC50 = 92 nM T70977 CFW9Q8 44448296 IC50 = 279 nM T70977 C4TFY7 44448297 IC50 = 630 nM T70977 CRS1Z9 44448298 IC50 = 200 nM T70977 CD3N2S 44448318 IC50 = 24 nM T70977 C54FTS 44448319 IC50 = 281 nM T70977 C4C2EM 44448320 IC50 = 49 nM T70977 C7JV9D 44448340 IC50 = 3500 nM T70977 CAK9P5 44448341 IC50 = 760 nM T70977 C2YK7C 44448342 IC50 = 180 nM T70977 C7Y1SX 44448360 IC50 = 960 nM T70977 CSE08W 44448362 IC50 = 490 nM T70977 CLCO97 44448363 IC50 = 4170 nM T70977 CNGP68 44448395 IC50 = 540 nM T70977 CK6WJ8 44448397 IC50 = 150 nM T70977 C3GK1N 44448430 IC50 = 4000 nM T70977 CML5S9 44448473 IC50 = 1700 nM T70977 C9KB0D 44448475 IC50 = 2900 nM T70977 CT7DU8 44448476 IC50 > 10000 nM T70977 CPZG30 44448478 IC50 = 2400 nM T70977 C8Z2ET 44448517 IC50 = 3500 nM T70977 C24CIE 44448518 IC50 = 1130 nM T70977 CT8A3E 44448519 IC50 = 3480 nM T70977 C3JFB4 44448552 IC50 = 3380 nM T70977 CWPD39 44448555 IC50 = 2990 nM T70977 CT86BF 44448556 IC50 = 3000 nM T70977 C29DPK 44448557 IC50 = 2610 nM T70977 C3SY5Z 44448591 IC50 = 1480 nM T70977 C5RJN6 44448630 IC50 = 1430 nM T70977 CCG8N5 44448663 IC50 = 1330 nM T70977 C6EZR8 44448678 IC50 = 1060 nM T70977 CP07GH 44448693 IC50 = 744 nM T70977 CT24RL 44448694 IC50 = 105 nM T70977 CX0QU1 44448695 IC50 = 169 nM T70977 C5A6US 44448701 IC50 = 890 nM T70977 CY0HI6 44448702 IC50 = 900 nM T70977 C0DV1I 44448703 IC50 = 860 nM T70977 C3ZHT1 44448715 IC50 = 51 nM T70977 C08EFA 44448716 IC50 = 75 nM T70977 C5S2AF 44448719 IC50 = 860 nM T70977 C38ASD 44448720 IC50 = 710 nM T70977 CK0S7D 44448735 IC50 = 26 nM T70977 CVA38F 44448737 IC50 = 477 nM T70977 C79YQL 44448738 IC50 = 23 nM T70977 CGP20A 44450492 IC50 = 18 nM T70977 CYV29J 44455333 IC50 > 15000 nM T70977 C8F0TR 44455389 IC50 = 30 nM T70977 C0NZK4 44455418 IC50 = 475 nM T70977 CKS5Y6 44455441 IC50 = 1585 nM T70977 CV2YT8 44455442 IC50 = 1628 nM T70977 C20YHS 44478652 IC50 = 81 nM T70977 CRG48I 44480699 IC50 = 94 nM T70977 C1US2Q 44480953 IC50 = 72 nM T70977 C03YLC 44480954 IC50 > 1000 nM T70977 CWK4F0 44480956 IC50 = 680 nM T70977 C30YRS 44481207 IC50 > 1000 nM T70977 CB3EA4 44481477 IC50 = 13 nM T70977 C31WOA 44482290 IC50 = 130 nM T70977 C03IGD 44540030 IC50 = 1584.89 nM T70977 C5LWU1 44540126 IC50 = 1258.93 nM T70977 CAT2R7 44540316 IC50 > 25118.86 nM T70977 C2T9GC 44540407 IC50 = 3162.28 nM T70977 CQ4PE7 44540492 IC50 = 7943.28 nM T70977 C4WRN5 44541014 IC50 = 5.9 nM T70977 C4AGX2 44550927 IC50 = 65000 nM T70977 C52TUH 44551057 IC50 > 10000 nM T70977 C3VRO9 44557921 IC50 > 10000 nM T70977 C5I3HT 44580807 IC50 = 8 nM T70977 CMH2A3 44580824 IC50 = 20 nM T70977 CTP7I4 44580861 IC50 = 20 nM T70977 C4JKW3 44581167 IC50 = 79 nM T70977 C9KG2I 44581261 IC50 = 1012 nM T70977 C5TBY3 44581605 IC50 = 1863 nM T70977 CEX34T 44581606 IC50 = 539 nM T70977 CROB85 44582642 IC50 = 0.35 nM T70977 CQ8W6D 44582643 IC50 = 23.8 nM T70977 CVL1D5 44582683 IC50 = 184 nM T70977 C3UIL7 44582684 IC50 = 0.95 nM T70977 C58JRZ 44582713 IC50 = 870 nM T70977 C9MQS1 44582714 IC50 = 1290 nM T70977 CJZ08I 44582715 IC50 = 4090 nM T70977 CN4RC3 44582716 IC50 = 260 nM T70977 CLFD52 44582743 IC50 = 7160 nM T70977 CWHR56 44582744 IC50 = 7.5 nM T70977 CZS9G7 44582745 IC50 = 0.51 nM T70977 C1S4WT 44582766 IC50 = 25.3 nM T70977 CAB2E1 44582767 IC50 = 48.3 nM T70977 CP5LO6 44582768 IC50 = 335 nM T70977 C0V6UM 44582789 IC50 = 88.7 nM T70977 CI4C5P 44582790 IC50 = 180 nM T70977 CT91FV 44582791 IC50 = 13.2 nM T70977 C9YB3M 44582816 IC50 = 710 nM T70977 COUV96 44582836 IC50 = 5.4 nM T70977 CL6JO8 44582837 IC50 = 5.1 nM T70977 C9MG0D 44582838 IC50 = 0.23 nM T70977 CP4X0U 44582855 IC50 = 0.73 nM T70977 CQ8F1K 44582856 IC50 = 10.2 nM T70977 CW2VP9 44582857 IC50 = 1.2 nM T70977 C1GU7V 44582871 IC50 = 314 nM T70977 CI96VH 44590237 IC50 = 54 nM T70977 C4CWG7 44590238 IC50 = 220 nM T70977 C5M4SW 44590239 IC50 = 94 nM T70977 CH7DA3 44590240 IC50 = 200 nM T70977 C39DYQ 44590241 IC50 = 280 nM T70977 CHD98A 44590242 IC50 = 91 nM T70977 CKR08B 44590275 IC50 = 68 nM T70977 C51VPS 44590376 IC50 = 630 nM T70977 C19DBV 44590377 IC50 = 13 nM T70977 C01UDJ 44590378 IC50 = 28 nM T70977 CT3NB5 44590379 IC50 = 5.7 nM T70977 C93MQS 44590380 IC50 = 340 nM T70977 CT95RZ 44590413 IC50 = 330 nM T70977 CC79SW 44590414 IC50 > 10000 nM T70977 CQDS96 44590415 IC50 = 680 nM T70977 CO1LP6 44590416 IC50 = 4.9 nM T70977 C95ZHC 44590463 IC50 = 16 nM T70977 CO1YT8 44590464 IC50 = 6.5 nM T70977 CLJ16E 44590465 IC50 = 18 nM T70977 C4EP3L 44590466 IC50 = 25 nM T70977 CFZM51 44590534 IC50 = 8.4 nM T70977 CZ3U0A 44590535 IC50 = 3.5 nM T70977 C74DZG 44590536 IC50 = 8.6 nM T70977 CI4BF2 44590537 IC50 = 2.5 nM T70977 CG2Y4Z 44590565 IC50 = 9.4 nM T70977 CP7C8O 44590595 IC50 > 10000 nM T70977 CLRZ35 44590756 IC50 = 7800 nM T70977 CQ80PN 44590760 IC50 = 13500 nM T70977 CV3QZ0 44590954 IC50 = 44 nM T70977 CCJE58 44590955 IC50 = 210 nM T70977 C5Z3LI 44591740 IC50 = 1900 nM T70977 COY57J 44592504 IC50 = 20000 nM T70977 CDN3C4 44622839 Ki = 1100 nM T70977 C5G0UA 44622840 Ki = 2100 nM T70977 C7PZ4E 44818424 IC50 = 1200 nM T70977 CG2E0J 44818425 IC50 = 13000 nM T70977 CQG2I1 44818426 IC50 > 10000 nM T70977 C6U2QM 44818427 IC50 > 10000 nM T70977 C4PQN9 44818428 IC50 > 10000 nM T70977 CQ0P8J 44818429 IC50 > 10000 nM T70977 CX9N2H 44818604 IC50 > 10000 nM T70977 C31LVM 44818605 IC50 > 10000 nM T70977 CY7X5Q 44818606 IC50 > 10000 nM T70977 CQ94CF 44818607 IC50 > 10000 nM T70977 CX8T3R 44818608 IC50 > 10000 nM T70977 CTV1Y5 44818609 IC50 > 10000 nM T70977 C7WEC0 44818784 IC50 > 100000 nM T70977 CR9XG5 44818785 IC50 = 700000 nM T70977 C5EZM6 44818786 IC50 > 10000 nM T70977 CHQT72 44818787 IC50 = 600000 nM T70977 CKGE16 44818788 IC50 > 10000 nM T70977 C1YFC4 44818789 IC50 > 1000000 nM T70977 CK49WN 45139234 IC50 = 860 nM T70977 CU3RF1 45139989 IC50 = 28 nM T70977 CQGZ06 45139991 IC50 = 48 nM T70977 CC2NT3 45267375 IC50 = 30600 nM T70977 CV45AE 45267376 IC50 = 660 nM T70977 C8BMT5 45267453 IC50 > 73340 nM T70977 C8Y9OZ 45267779 IC50 = 40 nM T70977 CNZ1Y6 45268307 IC50 = 960 nM T70977 C4UB5V 45268311 IC50 = 480 nM T70977 CWGA23 45268312 IC50 = 950 nM T70977 C5EBA2 45268316 IC50 = 750 nM T70977 C09TXA 45268667 IC50 = 30 nM T70977 C4Z0YO 45269184 IC50 = 550 nM T70977 C12PAK 45269191 IC50 = 1090 nM T70977 CIA8U1 45269192 IC50 = 12270 nM T70977 CM6ZI7 45269642 IC50 = 7 nM T70977 C87FEM 45270051 IC50 = 810 nM T70977 CK98GZ 45270062 IC50 = 22460 nM T70977 CCJ5S8 45270795 IC50 = 1140 nM T70977 C3L5JM 45270871 IC50 = 4890 nM T70977 CV04OL 45270879 IC50 = 3340 nM T70977 CPO6K5 45271266 Ki = 17 nM T70977 CIZ51Q 45271627 IC50 = 900 nM T70977 C1N7WA 45271725 IC50 = 310 nM T70977 C25KHF 45271869 IC50 = 6400 nM T70977 C8AC1S 45272193 IC50 = 2 nM T70977 CS27IJ 45272519 IC50 = 850 nM T70977 C6LB9J 45272589 IC50 = 2660 nM T70977 C4N2EH 45272601 IC50 = 13580 nM T70977 C5XL2N 45272602 IC50 = 2260 nM T70977 C8GUV9 45272605 IC50 = 12440 nM T70977 CMGS38 45272910 IC50 = 65 nM T70977 CP32VC 45273457 IC50 = 5690 nM T70977 C96TKH 45273503 IC50 = 12450 nM T70977 CXR29U 45273504 IC50 = 1790 nM T70977 CU53FK 45273505 IC50 = 260 nM T70977 CGA2K5 45482675 IC50 = 200 nM T70977 CUJS39 45482677 IC50 = 54 nM T70977 C4XOL3 45482681 IC50 = 50 nM T70977 CV48CZ 45482689 IC50 = 69 nM T70977 CFB31W 45482690 IC50 = 180 nM T70977 CI8G7M 45482691 IC50 = 790 nM T70977 CFD8I9 45482695 IC50 = 100 nM T70977 CMD8A5 45482696 IC50 = 140 nM T70977 C6E2SC 45482700 IC50 = 34 nM T70977 C39PSE 45482706 IC50 = 160 nM T70977 C14IQE 45482710 IC50 > 1000 nM T70977 CQG8R6 45482711 IC50 = 270 nM T70977 CGN0M3 45482715 IC50 = 200 nM T70977 CO7U1Y 45482716 IC50 > 1000 nM T70977 C0CG6J 45482717 IC50 = 190 nM T70977 C5LTU8 45482748 IC50 = 280 nM T70977 CM8XQ3 45482749 IC50 > 1000 nM T70977 CZXH74 45482750 IC50 = 20 nM T70977 CLZ5V4 45482754 IC50 = 110 nM T70977 CSLM96 45482758 IC50 = 66 nM T70977 C9HSZ2 45482759 IC50 = 35 nM T70977 CYJX54 45482760 IC50 = 42 nM T70977 CTM64G 45482765 IC50 = 35 nM T70977 CVZ19Q 45482766 IC50 = 38 nM T70977 C4YK2Z 45482767 IC50 = 77 nM T70977 C7GWS1 45482776 IC50 = 74 nM T70977 C73MDT 45482777 IC50 = 210 nM T70977 C6IR9X 45482948 IC50 > 10000 nM T70977 CDG6L4 45484160 IC50 = 486 nM T70977 CQ5SD4 46190876 IC50 = 160 nM T70977 CUA97D 46209401 IC50 = 500 nM T70977 CY3HW5 46224684 IC50 = 1300 nM T70977 CSWY60 46225572 IC50 = 260 nM T70977 CS9GL5 46225573 IC50 = 3860 nM T70977 CB5H9C 46225574 IC50 = 670 nM T70977 C8M1DT 46225589 IC50 = 64 nM T70977 C60XUQ 46226079 IC50 = 220 nM T70977 C5PCH8 46226080 IC50 = 470 nM T70977 C6UD1Y 46226095 IC50 > 10000 nM T70977 C7IF4T 46226096 IC50 = 280 nM T70977 CUDZ46 46226135 IC50 > 10000 nM T70977 C0P4CT 46226136 IC50 = 300 nM T70977 CPH49S 46226137 IC50 > 30000 nM T70977 CM5X8B 46226156 IC50 > 30000 nM T70977 C64TVL 46226417 IC50 = 210 nM T70977 C0BGH8 46227236 IC50 > 100000 nM T70977 C36SIO 46227237 IC50 > 100000 nM T70977 COJ9M1 46227238 IC50 > 100000 nM T70977 CR50QU 46227239 IC50 > 100000 nM T70977 C6QR3P 46227247 IC50 > 100000 nM T70977 C2H8AI 46227261 IC50 > 100000 nM T70977 CF4Z8V 46227308 IC50 = 5000 nM T70977 C7ON5A 46233287 IC50 = 358 nM T70977 CLSV86 46702565 Ki = 5800 nM T70977 CZS7O8 46843795 IC50 = 27000 nM T70977 C1U4NA 46843861 IC50 > 100000 nM T70977 CT03RU 46871676 IC50 = 8.5 nM T70977 CQB16A 46872415 Ki > 4000 nM T70977 CLS29B 46872626 IC50 > 10000 nM T70977 C3H0IG 46880254 IC50 = 2800 nM T70977 C24CMX 46880255 IC50 = 3100 nM T70977 C60KSN 46880256 IC50 = 8200 nM T70977 CW73FJ 46880257 IC50 = 220 nM T70977 C26SBC 46880299 IC50 = 31 nM T70977 CGUK43 46880300 IC50 = 6.4 nM T70977 C19QMX 46880301 IC50 = 35 nM T70977 CZ7X2O 46880302 IC50 = 1300 nM T70977 CIQW73 46880303 IC50 = 3.2 nM T70977 CNF9A5 46880334 IC50 = 8.2 nM T70977 CUYQ70 46880335 IC50 = 1.8 nM T70977 CGU86E 46880861 IC50 = 7 nM T70977 CZ36UN 46880908 IC50 = 2.4 nM T70977 CRW97F 46880909 IC50 = 6.6 nM T70977 C92JKU 46880910 IC50 = 22 nM T70977 CDX7O5 46880947 IC50 = 730 nM T70977 CQE90R 46880948 IC50 = 2000 nM T70977 CI23SC 46880949 IC50 = 350 nM T70977 CT46AI 46881730 IC50 > 10000000 nM T70977 CFDG95 46881822 IC50 = 17103 nM T70977 C6OM3Y 46881823 IC50 = 20532 nM T70977 C23IQK 46881852 IC50 = 25038 nM T70977 CQ7ET6 46881853 IC50 = 6 nM T70977 CDJ57I 46881879 IC50 = 12 nM T70977 C29PHE 46882055 IC50 = 4100 nM T70977 CNTS27 46883044 Ki = 380 nM T70977 C0DB5Z 46883045 Ki = 210 nM T70977 C9WE4S 46883122 Ki > 2500 nM T70977 CNTS75 46883123 Ki = 1000 nM T70977 CJS68B 46883124 Ki > 5000 nM T70977 CU3O2G 46883125 Ki > 5000 nM T70977 CH9RV4 46883165 Ki = 460 nM T70977 CT1K6A 46883166 Ki > 3300 nM T70977 CGZ1S4 46883167 Ki > 3300 nM T70977 C2VGJ9 46883168 Ki = 3200 nM T70977 CT5V8K 46883169 Ki > 3300 nM T70977 C2O8RZ 46886323 IC50 > 1000 nM T70977 CM8RX4 46886549 IC50 = 190 nM T70977 C70BLN 46886550 IC50 = 1570 nM T70977 CCV96R 46886665 IC50 = 1140 nM T70977 C3CRM0 46894040 IC50 = 169 nM T70977 C8RQ1Z 46902082 IC50 = 2000 nM T70977 C7LR8O 46902083 IC50 = 600 nM T70977 C1NKE3 46905987 IC50 = 3 nM T70977 C5OIK6 46918498 IC50 = 2500 nM T70977 CQR9K1 46933384 IC50 > 100000 nM T70977 C2B5XF 49765254 IC50 = 9600 nM T70977 CSO3H2 49788704 IC50 < 100 nM T70977 C6X1YA 49797869 IC50 = 3100 nM T70977 CHSF07 49806372 IC50 > 1000 nM T70977 CJZ5A0 49840306 IC50 > 10000 nM T70977 CB0S2P 49842666 IC50 > 100000 nM T70977 CO98FI 49843482 Ki = 58 nM T70977 CF91RS 49843531 IC50 > 10000 nM T70977 CT4ZN0 49855366 IC50 > 1000 nM T70977 C68DPT 49855367 IC50 = 534 nM T70977 CRTF14 49855368 IC50 = 53 nM T70977 C8QBE2 49855369 IC50 = 805 nM T70977 CZ06TP 49855370 IC50 > 1000 nM T70977 C58WDQ 49855371 IC50 = 314 nM T70977 C5CRH4 49855372 IC50 > 1000 nM T70977 C9X5YG 49855564 IC50 = 18 nM T70977 CIH3J2 49855565 IC50 = 7 nM T70977 C9LFE5 49855566 IC50 = 662 nM T70977 CXW1D8 49855567 IC50 = 710 nM T70977 CL5C4Y 49857866 IC50 = 17 nM T70977 CMS67Y 49857867 IC50 = 632 nM T70977 CECI61 49858058 IC50 > 1000 nM T70977 CAMH56 49858059 IC50 = 439 nM T70977 C4EWT7 49858060 IC50 = 247 nM T70977 C7OM5R 49858061 IC50 > 1000 nM T70977 CI48YQ 49858062 IC50 > 1000 nM T70977 CWZ8Q3 49858251 IC50 > 1000 nM T70977 C8GB5R 49858252 IC50 > 1000 nM T70977 C81VUI 49858253 IC50 = 855 nM T70977 C4VX7Q 49858254 IC50 = 671 nM T70977 CTW4G8 49858255 IC50 > 1000 nM T70977 C1MQ3C 49858256 IC50 = 719 nM T70977 C23QZC 49858257 IC50 = 811 nM T70977 CV34FE 49858258 IC50 > 1000 nM T70977 CV7GB4 49863015 IC50 = 365 nM T70977 C6WB4Z 49863065 IC50 = 781 nM T70977 CD67FY 49863104 IC50 > 20000 nM T70977 C83VHI 49864785 IC50 > 100000 nM T70977 C2UTK6 49864850 IC50 > 100000 nM T70977 CAE53W 49865153 IC50 > 100000 nM T70977 CQE9D1 50925411 IC50 = 3 nM T70977 C2Y6QS 50938552 IC50 > 10000 nM T70977 C0CF5H 50993749 IC50 = 780 nM T70977 C12NOU 50993750 IC50 = 670 nM T70977 C58CUD 50993751 IC50 = 4080 nM T70977 CG7MI0 50993752 IC50 = 2260 nM T70977 CM42BY 51000510 Ki = 20 nM T70977 CAZQ43 51003133 IC50 > 1000 nM T70977 C9NYP4 51036677 IC50 > 10000 nM T70977 C4WRY3 51037112 IC50 > 10000 nM T70977 CRI28Z 51037948 IC50 > 10000 nM T70977 CA7M0O 51038938 IC50 = 1300 nM T70977 CEL8V6 51038948 IC50 = 4100 nM T70977 CCQ1U2 51038949 IC50 = 1000 nM T70977 CSB93C 51038950 IC50 = 1600 nM T70977 CI8W0M 51038951 IC50 = 2000 nM T70977 CP2XG0 51038952 IC50 = 900 nM T70977 C32FZW 51038953 IC50 = 600 nM T70977 CZSG50 51038954 IC50 = 500 nM T70977 CQ1ZC6 51038965 IC50 = 1200 nM T70977 C8MJW7 51038968 IC50 = 1200 nM T70977 C3UVM4 51038970 IC50 = 300 nM T70977 C96EIN 51038980 IC50 = 900 nM T70977 CJEW87 51038995 IC50 = 300 nM T70977 C6M9TQ 51039273 IC50 = 3300 nM T70977 CR8AC5 51185962 IC50 = 131 nM T70977 CDU4Q5 51346827 Ki = 446 nM T70977 CP89UE 51346932 IC50 = 6.1 nM T70977 CQ5G2F 51346933 IC50 = 17.4 nM T70977 CS7Q3D 51347384 IC50 > 100000 nM T70977 C16UXT 51347682 IC50 = 50000 nM T70977 CJU19H 51347839 IC50 = 4000 nM T70977 CE9TJ5 51347987 IC50 = 8100 nM T70977 CT9F5Q 51352270 IC50 = 36 nM T70977 CEQN27 52936621 Ki > 1000 nM T70977 CM24LF 52938983 IC50 = 2.73 nM T70977 C65ZXV 52949623 IC50 = 638 nM T70977 C71BOQ 52952011 IC50 = 3000 nM T70977 CKU14E 53237693 IC50 = 152 nM T70977 CJ56EO 53244398 IC50 = 9 nM T70977 C64IQX 53244399 IC50 = 40 nM T70977 C1P3BC 53244475 IC50 = 215 nM T70977 CRQ6B1 53245729 IC50 = 125.89 nM T70977 CI2QX4 53245730 IC50 = 158.49 nM T70977 C8T3NL 53245731 IC50 = 125.89 nM T70977 C6OTY5 53251320 IC50 > 30000 nM T70977 CYS65F 53262860 IC50 = 5 nM T70977 CWU12F 53262861 IC50 = 47 nM T70977 C3YQR9 53308827 IC50 = 890 nM T70977 C0TLX7 53310972 IC50 = 13400 nM T70977 CS14NJ 53310974 IC50 > 10000 nM T70977 CKA60L 53310975 IC50 = 580 nM T70977 C5UWF0 53310976 IC50 = 4470 nM T70977 C4MR7F 53317124 IC50 > 894 nM T70977 C3I2LV 53317125 IC50 = 84.1 nM T70977 CJA71P 53317758 IC50 = 537 nM T70977 CF7D3J 53317876 IC50 = 1975 nM T70977 CR20TC 53318412 IC50 > 9000 nM T70977 CQ5TI1 53318413 IC50 = 115 nM T70977 CZS8K4 53319042 Ki = 1298 nM T70977 C51JLM 53319742 IC50 = 62 nM T70977 CO8ZA4 53319743 IC50 > 731 nM T70977 C9GH0Q 53319744 IC50 = 133 nM T70977 C15HNX 53320116 IC50 > 592 nM T70977 CUD21V 53320263 Ki = 528 nM T70977 CZLW74 53320503 IC50 = 1270 nM T70977 C5V6SK 53322383 IC50 = 51 nM T70977 CESA85 53323614 Ki = 891 nM T70977 CELV57 53323742 IC50 > 10000 nM T70977 COM58A 53324306 IC50 = 233 nM T70977 C2W9OA 53324451 IC50 > 10000 nM T70977 CP58BQ 53324485 IC50 = 325 nM T70977 CVA13E 53325012 IC50 > 401 nM T70977 C0OY2V 53325013 IC50 = 62.8 nM T70977 CYW98L 53326306 IC50 = 50.1 nM T70977 C0SWH5 53348216 IC50 > 40000 nM T70977 C8ZRE3 53356518 IC50 > 50000 nM T70977 CBH27E 53361525 IC50 = 22450 nM T70977 CA2DU1 53363044 IC50 = 9950 nM T70977 CG50TB 53380598 IC50 = 79.43 nM T70977 CC8G2I 53380599 IC50 = 630.96 nM T70977 C8NA4L 53384644 IC50 > 30000 nM T70977 C71OXL 53388145 IC50 = 140000 nM T70977 CDL28G 53388146 IC50 = 510000 nM T70977 CAI80C 53484135 IC50 = 44 nM T70977 C8CVT6 53628878 IC50 = 7.8 nM T70977 C9G8UO 53628896 IC50 = 13 nM T70977 C6AUQ2 53628921 IC50 = 1500 nM T70977 CSW32F 54581340 IC50 = 45 nM T70977 CB1MX5 54676647 IC50 = 4500 nM T70977 C7F6XB 54676762 IC50 = 7300 nM T70977 CYM1C7 54682955 IC50 > 20000 nM T70977 C0OQR4 54683111 IC50 = 8700 nM T70977 CDT3J9 54684571 IC50 > 20000 nM T70977 CS05IU 54687035 IC50 > 20000 nM T70977 CBU9T3 54687079 IC50 > 20000 nM T70977 CVT01A 54687084 IC50 = 4500 nM T70977 C16UOP 54687085 IC50 = 3010 nM T70977 CWG3V0 54696404 IC50 > 20000 nM T70977 C5QTJ7 54705584 IC50 > 20000 nM T70977 C2G3AY 54726684 IC50 = 1900 nM T70977 CC4S8H 54728388 IC50 > 100000 nM T70977 CAI3H8 54728389 IC50 = 25000 nM T70977 CE1ZK6 54759168 IC50 > 10000 nM T70977 C1XS2J 54760383 IC50 > 10000 nM T70977 C4S1HX 56589672 IC50 = 12 nM T70977 CUH6T9 56603827 IC50 = 13 nM T70977 CN9QD7 56643097 IC50 = 79.43 nM T70977 CS87BO 56658164 IC50 = 560 nM T70977 C4O1WR 56660107 IC50 = 19.95 nM T70977 C4XSR0 56661674 IC50 = 75 nM T70977 C1LM7F 56661675 IC50 = 49 nM T70977 CD6V3U 56662952 IC50 > 50000 nM T70977 C91IHZ 56663572 IC50 = 316.23 nM T70977 CIT3C7 56664963 IC50 = 3400 nM T70977 CJXG57 56665083 IC50 = 1500 nM T70977 C8J6EP 56665084 IC50 = 31 nM T70977 CDK9G2 56665085 IC50 = 440 nM T70977 CD7P2G 56665389 IC50 = 110 nM T70977 CGLN74 56666429 IC50 = 500 nM T70977 C0O2EN 56667018 IC50 = 2511.89 nM T70977 C4Z2YU 56667019 IC50 = 3981.07 nM T70977 CIM94L 56668847 IC50 = 3640000 nM T70977 CQ74RS 56670463 IC50 = 316.23 nM T70977 CGV6Y1 56671901 IC50 = 2100 nM T70977 CH4F0C 56671902 IC50 = 17000 nM T70977 CQX68C 56672039 IC50 = 16000 nM T70977 CWV70H 56673950 IC50 = 12.59 nM T70977 CJA6E7 56675282 IC50 = 26000 nM T70977 CP0OY1 56675417 IC50 = 160 nM T70977 C8PK0W 56675716 IC50 = 1430000 nM T70977 CQ1OT2 56677279 IC50 = 10 nM T70977 C7ID8C 56677280 IC50 = 158.49 nM T70977 C5L3ZE 56678608 IC50 = 1200 nM T70977 CIH6W2 56678997 IC50 = 98 nM T70977 CU1GX5 56680583 IC50 = 251.19 nM T70977 COM4F3 56680584 IC50 = 10000 nM T70977 CVLW80 56683909 IC50 = 501.19 nM T70977 C2MQ6I 56683910 IC50 = 10 nM T70977 CDP30U 56683911 IC50 = 12.59 nM T70977 CA7T5R 56683912 IC50 = 125.89 nM T70977 C4Z0OC 56834890 IC50 = 180 nM T70977 C67TJQ 56834891 IC50 = 340 nM T70977 CBOD63 56835089 IC50 > 30000 nM T70977 CR4H3M 56835099 IC50 = 490 nM T70977 CP8T5I 56835100 IC50 > 30000 nM T70977 CR3YN1 56945119 IC50 = 0.6 nM T70977 CR16SD 56947170 IC50 = 70 nM T70977 C6HOV4 56950795 IC50 = 0.57 nM T70977 CPI3O8 56962315 Ki = 20 nM T70977 CRVZ25 56964906 IC50 = 4600 nM T70977 CPHX64 57325478 IC50 > 50000 nM T70977 CQ9BW4 57325479 IC50 > 50000 nM T70977 COU15Y 57326116 IC50 = 7000 nM T70977 CJ3EV5 57326117 IC50 = 1800 nM T70977 CYB1E4 57326217 IC50 = 1400 nM T70977 CELU72 57326220 IC50 = 2000 nM T70977 CU7YP0 57326223 IC50 = 1000 nM T70977 C83YSU 57326315 IC50 = 300 nM T70977 CXIG75 57326316 IC50 = 1100 nM T70977 CR46JC 57326399 IC50 = 800 nM T70977 CU3AK2 57326494 IC50 = 1100 nM T70977 CHW02R 57328617 IC50 = 7 nM T70977 CJ73IL 57328618 IC50 = 6 nM T70977 C9ZMN6 57328619 EC50 = 100 nM T70977 C8X5JG 57384039 IC50 = 130 nM T70977 C5KM9Z 57391251 IC50 = 1.4 nM T70977 CXNS85 57391252 IC50 = 150 nM T70977 CZ1WP8 57391298 IC50 = 316.23 nM T70977 CAE9H8 57391299 IC50 = 3162.28 nM T70977 CZ1C4U 57391300 IC50 = 63095.73 nM T70977 C5GPR2 57391376 EC50 = 3900 nM T70977 C35FGD 57391377 EC50 = 21000 nM T70977 C29PXR 57393017 IC50 = 16 nM T70977 CZ45KW 57393077 IC50 = 251.19 nM T70977 C2RV8M 57393078 IC50 = 31622.78 nM T70977 CXA72Y 57393079 IC50 = 1995.26 nM T70977 C8SJ1W 57393133 EC50 = 230 nM T70977 C2PW9N 57393134 IC50 = 31 nM T70977 CRC23Y 57393135 EC50 = 240 nM T70977 CLPN10 57393136 IC50 = 8 nM T70977 CN90ST 57393137 IC50 = 10 nM T70977 C1O5PX 57394800 IC50 = 6309.57 nM T70977 CYV54G 57394801 IC50 = 2511.89 nM T70977 C3SGR9 57394802 IC50 = 7943.28 nM T70977 CS85QL 57394803 IC50 = 31622.78 nM T70977 C9L2SB 57394812 IC50 = 31.62 nM T70977 CD6Y9Z 57395116 IC50 > 30000 nM T70977 C8W6IG 57395117 IC50 > 30000 nM T70977 CW56FQ 57396415 IC50 = 71 nM T70977 C12CXP 57396561 IC50 = 316.23 nM T70977 CQI0X9 57396562 IC50 = 31.62 nM T70977 CBTP07 57396563 IC50 = 398.11 nM T70977 CJ6NV4 57396564 IC50 = 1258.93 nM T70977 CK3FP5 57396565 IC50 = 79.43 nM T70977 CKE3B0 57396576 IC50 = 100 nM T70977 CX17PL 57396577 IC50 = 19.95 nM T70977 CY4E8K 57396633 EC50 = 2700 nM T70977 CG7S0D 57396882 IC50 > 30000 nM T70977 CVQK90 57397197 IC50 = 1800 nM T70977 C9MLJ4 57398214 IC50 = 140 nM T70977 CIBF21 57398344 IC50 > 25118.86 nM T70977 CF23NI 57398345 IC50 = 630.96 nM T70977 CI5GW3 57398346 IC50 = 3162.28 nM T70977 CYR9E5 57398347 IC50 = 12.59 nM T70977 C8B3PI 57398348 IC50 = 19.95 nM T70977 C0CQ6Y 57398403 IC50 = 2000 nM T70977 C9H8AR 57398404 IC50 = 2800 nM T70977 C0XTH3 57398405 EC50 = 13 nM T70977 C96WSN 57398406 EC50 = 95 nM T70977 CELC82 57398900 IC50 = 6300 nM T70977 CI76LU 57399379 IC50 = 9500 nM T70977 C8R7ES 57399952 IC50 = 0.86 nM T70977 C5CLX0 57400013 IC50 = 1995.26 nM T70977 CB7EC9 57401736 IC50 = 40 nM T70977 CX8V3C 57401737 IC50 = 67 nM T70977 CR4OA1 57401810 IC50 = 1995.26 nM T70977 C0GL5D 57401811 IC50 = 3162.28 nM T70977 C2YZE6 57401822 IC50 = 31.62 nM T70977 C3G4QA 57401875 IC50 = 140 nM T70977 CXC2R0 57401876 EC50 = 400 nM T70977 CE12CQ 57402393 IC50 = 2600 nM T70977 CQ3A5B 57402394 IC50 = 2800 nM T70977 C7STM0 57403370 IC50 = 1 nM T70977 CO13ZS 57403371 IC50 = 10 nM T70977 CUT03F 57403459 IC50 = 33 nM T70977 CC4P3A 57403470 IC50 = 180 nM T70977 CSPB30 57403520 IC50 = 251.19 nM T70977 C5OQA0 57403528 IC50 = 19.95 nM T70977 CHV6R9 57403529 IC50 = 630.96 nM T70977 CH0L5I 57403589 EC50 = 310 nM T70977 C8P6RD 57505528 IC50 > 10000 nM T70977 CFZ40T 57522594 IC50 = 172 nM T70977 CEW5L7 57522817 IC50 = 22 nM T70977 C4SEH5 57522818 IC50 = 316 nM T70977 CF8IP6 57522819 IC50 < 5 nM T70977 CJ56CE 57522820 IC50 = 185 nM T70977 C3XI2P 57523093 IC50 = 233 nM T70977 CUH3B5 57523094 IC50 = 758 nM T70977 C3QF2X 57523095 IC50 = 129 nM T70977 C9M0AE 57593933 IC50 = 2.3 nM T70977 C29XDT 57593994 IC50 = 4.3 nM T70977 C5WH0O 57594057 IC50 = 630 nM T70977 CAC7U3 57594088 IC50 = 4.3 nM T70977 C3BH2O 57766675 EC50 = 10 nM T70977 C6GRC3 57766676 IC50 = 3 nM T70977 CPN18I 57766724 IC50 = 17 nM T70977 C0UOQ3 57766728 IC50 = 2 nM T70977 C9W5GF 57766769 EC50 = 62 nM T70977 C1BG5X 57766788 EC50 = 150 nM T70977 CC3YH6 57766798 IC50 = 3 nM T70977 CHU61A 57766836 EC50 = 1.5 nM T70977 CA30DY 57766848 IC50 = 9 nM T70977 CD01ZI 57766857 IC50 = 1 nM T70977 C3ZQM6 57766873 EC50 = 9 nM T70977 CP1G6T 57766887 EC50 = 130 nM T70977 C5XRP3 57766899 EC50 = 310 nM T70977 C4Z2QK 57766920 EC50 = 80 nM T70977 CZBL29 57766931 IC50 = 10 nM T70977 C3K6JN 57766969 EC50 = 10 nM T70977 C1B7US 57766970 EC50 = 10 nM T70977 C8I2JX 57798425 IC50 = 0.47 nM T70977 C52UJG 57798468 IC50 = 13 nM T70977 C0JCN7 57798480 IC50 = 4.6 nM T70977 CLYT61 57798492 IC50 = 0.87 nM T70977 CO7C9R 57798603 IC50 = 2.9 nM T70977 C0VU2Z 57798682 IC50 = 0.23 nM T70977 C1QX8T 57798887 IC50 = 3.2 nM T70977 C4K8HW 57834331 IC50 > 10000 nM T70977 CRI32E 57869872 IC50 > 1000 nM T70977 CO1B7C 57869916 IC50 = 4.2 nM T70977 C7YO6F 57869935 IC50 = 43 nM T70977 C9OBT1 57869953 IC50 = 3.8 nM T70977 CD9XV0 57869954 IC50 = 3.9 nM T70977 C4R6NA 57870014 IC50 = 2.7 nM T70977 C2H8ZW 57870102 IC50 = 14 nM T70977 C7C4VE 57870158 IC50 = 4.1 nM T70977 C2CR3O 57870171 IC50 = 1.2 nM T70977 CTW61H 57870208 IC50 = 24 nM T70977 C1W3IG 57877690 IC50 = 903 nM T70977 CHB6L1 57877715 IC50 = 2466 nM T70977 C0QFL3 57877765 IC50 = 7.4 nM T70977 CWI7T3 57877786 IC50 = 430 nM T70977 CFCG71 57877807 IC50 = 791 nM T70977 C6BPR2 58985201 IC50 > 50000 nM T70977 CT3EW2 59292007 IC50 = 980 nM T70977 CON8H1 59326984 IC50 = 30800 nM T70977 C1YTI8 59472018 Ki = 22 nM T70977 C4S6HC 59581274 IC50 = 12300 nM T70977 CXJ63M 59603829 IC50 = 84 nM T70977 CQEU96 59603842 IC50 = 23 nM T70977 C2P3CW 59793866 IC50 = 27 nM T70977 CGOF90 59793923 IC50 = 77 nM T70977 C2C0GV 59793933 IC50 = 13 nM T70977 C2W1TF 60001863 IC50 = 51 nM T70977 COH62U 60097413 IC50 > 3300 nM T70977 C1MR8Q 60097495 IC50 > 2500 nM T70977 CB1K7F 60147995 IC50 = 42180 nM T70977 CES0Y6 60147996 IC50 = 35680 nM T70977 CK6WO0 66552478 IC50 < 10000 nM T70977 C1M4OI 66553053 IC50 = 107 nM T70977 CIM7H1 66575095 IC50 = 10800 nM T70977 CF15KL 66771109 IC50 = 2.2 nM T70977 C1HSE0 67035086 IC50 = 1800 nM T70977 CWI6K5 67035106 IC50 > 10000 nM T70977 C37NKO 67129970 IC50 > 10000 nM T70977 CK80LJ 67130050 IC50 > 10000 nM T70977 C0ZLN2 68160176 IC50 = 200 nM T70977 C8I7GC 68293638 IC50 > 10000 nM T70977 CD56XK 68293660 IC50 > 10000 nM T70977 C7GRV2 68755406 IC50 > 10000 nM T70977 C0HA8V 68783839 IC50 = 34 nM T70977 CJVI10 68882695 IC50 = 0.64 nM T70977 C5DGR9 69036886 IC50 = 2988 nM T70977 CEI1T7 69545106 IC50 > 10000 nM T70977 CO58CT 69643651 Ki = 120 nM T70977 CS7AK8 69644160 Ki = 300 nM T70977 C1NCF3 69911184 IC50 > 10000 nM T70977 C4GJ0V 70682029 EC50 = 23 nM T70977 C4TM6F 70682212 IC50 = 1400 nM T70977 C9PE4T 70682214 IC50 = 6000 nM T70977 CNKB34 70682366 IC50 = 166 nM T70977 CW4C1K 70684312 IC50 = 1000 nM T70977 CGXQ82 70686290 EC50 = 10 nM T70977 C7OX5Z 70686473 IC50 = 700 nM T70977 C2MPQ3 70686838 IC50 = 44500 nM T70977 C2GS7T 70688399 IC50 = 47 nM T70977 C16PHW 70690441 IC50 = 30 nM T70977 CZ91YU 70690442 EC50 = 20 nM T70977 COM2C3 70690671 IC50 = 2170 nM T70977 C0RT2G 70690776 IC50 = 86 nM T70977 CCJH52 70691010 IC50 = 30800 nM T70977 CAJF37 70693140 IC50 = 24200 nM T70977 C2U7ES 70693141 IC50 = 30100 nM T70977 CQ75AH 70693142 IC50 = 60000 nM T70977 CLK38P 70693934 IC50 = 2100 nM T70977 C2XV4Q 70694953 IC50 = 36 nM T70977 CSX6M5 70696681 EC50 = 300 nM T70977 CP08FT 70696865 IC50 = 2600 nM T70977 C1IEJ2 70789254 IC50 = 138000 nM T70977 C8T7ZP 70789255 IC50 = 55000 nM T70977 CH0B8N 70789756 IC50 > 30000 nM T70977 CL1HY5 71212233 IC50 = 1995 nM T70977 CKX52R 71212291 IC50 = 225 nM T70977 C0T2VB 71212317 IC50 = 14 nM T70977 C5B8NS 71212337 IC50 = 164 nM T70977 CSN04E 71212395 IC50 = 127 nM T70977 C1OCW0 71212403 IC50 = 176 nM T70977 CBX2I4 71212419 IC50 = 234 nM T70977 CLS4R3 71212434 IC50 = 153 nM T70977 CTF8M7 71212446 IC50 = 32 nM T70977 C2Z8CX 71212514 IC50 = 84 nM T70977 CBT7L3 71212517 IC50 = 966 nM T70977 C7VA0I 71450358 IC50 > 62500 nM T70977 CZ96WN 71450733 IC50 > 100000 nM T70977 C7NS3P 71450734 IC50 > 100000 nM T70977 CPVN07 71451532 Ki > 1000000 nM T70977 C0U7AH 71451533 Ki = 10 nM T70977 CZ2OE6 71452173 IC50 = 1.491 nM T70977 CSPN93 71452174 IC50 = 1220 nM T70977 CR53ZS 71452175 IC50 = 7830 nM T70977 CM14JZ 71452176 IC50 = 38100 nM T70977 CEBO91 71452977 IC50 > 10000 nM T70977 C19EDO 71453604 Ki = 0.99 nM T70977 CX1KZ0 71453985 IC50 = 25600 nM T70977 C0N3HU 71455067 Ki = 20 nM T70977 CFGP02 71455731 IC50 > 30000 nM T70977 CKT60L 71455860 Ki = 102 nM T70977 CVG56J 71456067 IC50 = 25000 nM T70977 C9EK2X 71456068 IC50 = 47500 nM T70977 CINV12 71456867 Ki = 5800 nM T70977 CT4SB5 71456868 Ki = 1600 nM T70977 CS27GC 71457514 IC50 = 16 nM T70977 C16OVY 71457515 IC50 > 62500 nM T70977 CRL8H2 71457865 IC50 = 480000 nM T70977 C4GT3W 71457866 IC50 > 100000 nM T70977 CY6WI2 71458575 IC50 = 330 nM T70977 CHQZ25 71459584 IC50 > 10000 nM T70977 CYFO01 71459782 IC50 = 40000 nM T70977 C3KIM9 71461149 IC50 = 98 nM T70977 C9AJH5 71462252 Ki > 1000000 nM T70977 CW6MK4 71462888 IC50 = 1120 nM T70977 C9V6KY 71462889 IC50 = 4000 nM T70977 C9Z8AP 71543313 IC50 = 1780 nM T70977 C31POA 71547418 IC50 = 9000 nM T70977 CAR40E 71547419 IC50 = 3120 nM T70977 C0Z9GS 71547420 IC50 = 5800 nM T70977 CK62WS 71547496 IC50 > 20000 nM T70977 C1A5ZX 71547498 IC50 = 5250 nM T70977 C1C5EM 71547499 IC50 = 5510 nM T70977 CQ4NZ7 71547500 IC50 = 3540 nM T70977 C7I8MJ 71547501 IC50 = 3810 nM T70977 C97SEY 71547575 IC50 = 6280 nM T70977 CR1U2B 71547576 IC50 = 4280 nM T70977 C9KLW5 71547577 IC50 = 7340 nM T70977 CR6ZA8 71547578 IC50 = 2010 nM T70977 C0P8UA 71547579 IC50 = 8480 nM T70977 CD0BQ8 71547580 IC50 = 5950 nM T70977 CUBZ39 71547653 IC50 = 9420 nM T70977 C5TC0V 71547655 IC50 = 6660 nM T70977 CW6H7M 71547656 IC50 = 4030 nM T70977 CMI60Z 71547657 IC50 = 4830 nM T70977 C9R4JU 71547735 IC50 = 5960 nM T70977 CB2U9W 71547736 IC50 = 5990 nM T70977 CCN01X 71547862 IC50 > 10000 nM T70977 CA3O6K 71552696 IC50 = 1680 nM T70977 C1NPL0 71552941 IC50 > 30000 nM T70977 CA4PS8 71552942 IC50 > 30000 nM T70977 C3UA9C 71553011 IC50 = 30000 nM T70977 CEZ15Y 71553012 IC50 = 30000 nM T70977 CVIA91 71553085 IC50 = 30000 nM T70977 C1TR3O 71553152 IC50 = 30000 nM T70977 C6S1YB 71578237 IC50 > 100000 nM T70977 CZRG18 71578238 IC50 > 100000 nM T70977 C0W8OF 71578239 IC50 > 100000 nM T70977 CJ7H2N 71578240 IC50 > 100000 nM T70977 CHY91V 71578307 IC50 = 90 nM T70977 CIY6J3 71578308 IC50 > 100000 nM T70977 C1I5DW 71578309 IC50 = 73900 nM T70977 C5I9DH 71578310 IC50 = 76100 nM T70977 CIB67H 71578311 IC50 = 73700 nM T70977 CK9QJ2 71578312 IC50 > 100000 nM T70977 CD6XH7 71578313 IC50 = 27800 nM T70977 C0W2KX 71578373 IC50 = 27 nM T70977 C6TX9R 71578374 IC50 = 29 nM T70977 C2D1RN 71578375 IC50 = 86 nM T70977 CBN0W4 71578376 IC50 = 37800 nM T70977 CG08YE 71578377 IC50 = 23000 nM T70977 CCSL65 71578378 IC50 = 81500 nM T70977 CMXQ32 71578379 IC50 = 71000 nM T70977 C2YS0T 71578380 IC50 = 67800 nM T70977 C73MEW 71578445 IC50 = 75 nM T70977 C5NH3V 71578446 IC50 = 195 nM T70977 CC65WU 71578447 IC50 = 164 nM T70977 CIP6Q2 71578520 IC50 = 56 nM T70977 CPJ19D 71578658 IC50 = 35 nM T70977 C5W0GC 71578744 IC50 = 19 nM T70977 CLZ59B 71578745 IC50 = 17 nM T70977 CZ31PU 71583657 IC50 > 10000 nM T70977 C4OJP2 71680627 IC50 = 310 nM T70977 C67EFA 71714627 IC50 = 870 nM T70977 CL60MW 71714628 IC50 = 31 nM T70977 CH4I5P 71714649 IC50 = 72 nM T70977 CQV5M6 71714651 IC50 = 1400 nM T70977 C35ZQM 71714654 IC50 = 230 nM T70977 C0HUG5 71714668 IC50 = 27 nM T70977 C8RKD7 71714669 IC50 = 18 nM T70977 CJ2FX3 71714670 IC50 = 541 nM T70977 CMIL20 71714698 IC50 = 580 nM T70977 CSGK93 71714699 IC50 = 750 nM T70977 C7YD3C 71714700 IC50 = 1510 nM T70977 CZ4Q8C 71714701 IC50 = 1130 nM T70977 C6I7RC 71714702 IC50 = 530 nM T70977 C4HE7Z 71715678 IC50 = 350 nM T70977 CAQY29 71720048 IC50 = 40000 nM T70977 C28CUD 71733640 IC50 = 148 nM T70977 C5C2LF 71733641 IC50 = 114 nM T70977 CZF2L8 71733644 IC50 = 3.7 nM T70977 C7MNY1 71733646 IC50 = 11.5 nM T70977 C5S8JB 71733737 IC50 = 0.2 nM T70977 CPV57E 71733739 IC50 = 0.59 nM T70977 C04YBL 71733740 IC50 = 1.9 nM T70977 CV74XJ 71733742 IC50 = 0.53 nM T70977 C8KOH4 71733835 IC50 = 0.013 nM T70977 C7R1MY 71734778 IC50 = 21.4 nM T70977 CZ0IS2 71734779 IC50 = 4.8 nM T70977 C4D0RQ 71734780 IC50 = 15 nM T70977 CS9NP7 71734853 IC50 = 116 nM T70977 C56VRS 71734855 IC50 = 41.1 nM T70977 CN9OP4 71734857 IC50 = 404 nM T70977 C7S6UM 71734859 IC50 = 202 nM T70977 CW3Q9I 71734860 IC50 = 19.8 nM T70977 C05JPQ 71734933 IC50 = 39.7 nM T70977 C91RMV 71734934 IC50 = 82.3 nM T70977 CY9LW5 71734935 IC50 = 35.7 nM T70977 C57WPJ 71734936 IC50 = 5.3 nM T70977 CT7H6A 71734937 IC50 = 25.2 nM T70977 CPLR89 71734938 IC50 = 17.6 nM T70977 CN21QA 71735022 IC50 = 58.2 nM T70977 CW5C7R 71735023 IC50 = 65.9 nM T70977 C7NH5U 71735024 IC50 = 127 nM T70977 C32NZT 71735026 IC50 = 5.3 nM T70977 CK09EO 71735028 IC50 = 0.87 nM T70977 C8D0CB 71735029 IC50 = 11.2 nM T70977 C5DTG3 72696513 IC50 = 4608 nM T70977 CE1VB4 72696779 IC50 = 386 nM T70977 C0DL3F 72698602 IC50 = 7.77 nM T70977 C5G6VX 72708285 IC50 = 960 nM T70977 CVHW25 72708286 IC50 = 1290 nM T70977 CPQ6L1 72708287 IC50 = 680 nM T70977 C8SJ0F 72708790 IC50 = 460 nM T70977 C24RKQ 72708826 IC50 = 8840 nM T70977 C2XZW3 72708899 IC50 = 360 nM T70977 CKN46T 72708901 IC50 = 380 nM T70977 CZT13L 72708902 IC50 = 1900 nM T70977 C4B5RW 72725141 IC50 = 272 nM T70977 C5N8JY 72725258 IC50 = 9800 nM T70977 CI9B8V 72725478 IC50 = 6.5 nM T70977 C5FO1K 73333976 IC50 = 1.1 nM T70977 C2AG9F 73425095 IC50 = 7960 nM T70977 CVF5P0 73603034 IC50 = 23000 nM T70977 CT14IJ 75009054 IC50 = 13 nM T70977 CKN4F7 76313996 IC50 = 810 nM T70977 C5ZHE6 76317537 IC50 = 1000 nM T70977 C85TUR 76321270 IC50 = 1210 nM T70977 CA8OD1 76321272 IC50 = 940 nM T70977 CLYH23 76328447 IC50 = 690 nM T70977 CO9HK4 76328448 IC50 = 440 nM T70977 C5IOT9 76331317 IC50 = 120 nM T70977 C7AWU4 76332128 IC50 = 240 nM T70977 CJ2T9E 76332983 IC50 > 10000 nM T70977 CRE2U3 77050682 IC50 = 690 nM T70977 CP89YE 77939322 IC50 > 10000 nM T70977 CI6NP8 82276586 IC50 > 10000 nM T70977 CPG3A5 86302574 IC50 = 16184 nM T70977 C2ME7Y 86340067 IC50 = 6050 nM T70977 C1HW4B 89735655 IC50 = 150 nM T70977 C74PMG 89767064 IC50 = 5170 nM T70977 COM1K4 89767067 IC50 = 360 nM T70977 CE6M3J 89767087 IC50 = 400 nM T70977 CL9Y8B 89767178 IC50 = 70 nM T70977 C8W7ZM 89767184 IC50 = 12 nM T70977 CWEF34 89767201 IC50 = 300 nM T70977 C70NDL 89767207 IC50 = 50 nM T70977 CHGR80 89767213 IC50 = 490 nM T70977 CSXU34 89767287 IC50 = 2100 nM T70977 CF76RG 89767293 IC50 = 40 nM T70977 CYB09J 89767319 IC50 = 360 nM T70977 CY8FT0 89767330 IC50 = 320 nM T70977 C9U1DW 89767350 IC50 = 270 nM T70977 CD16QO 89767382 IC50 = 260 nM T70977 CONQ18 89767395 IC50 = 21 nM T70977 CJM26X 89767412 IC50 = 330 nM T70977 CQB96V 89767420 IC50 = 130 nM T70977 CE3F1O 89767466 IC50 = 9.6 nM T70977 CVWZ64 89767472 IC50 = 230 nM T70977 C4NI9C 89767523 IC50 = 17 nM T70977 C5CW0U 89767636 IC50 = 6 nM T70977 CXA59K 89767659 IC50 = 950 nM T70977 CW0U2T 89768926 IC50 = 670 nM T70977 C2LK4O 89777800 IC50 = 400 nM T70977 C1CA9S 89777804 IC50 = 360 nM T70977 CDS9Z5 89777805 IC50 = 1400 nM T70977 C3ER8P 89777807 IC50 = 640 nM T70977 CYF1Q8 89777931 IC50 = 250 nM T70977 CKO03E 89777934 IC50 = 790 nM T70977 CC2AY5 89777935 IC50 = 580 nM T70977 CWS6J4 89777943 IC50 = 45 nM T70977 CWLH32 89777944 Ki = 600 nM T70977 CZ0N2G 89777945 IC50 = 200 nM T70977 CX0W9Z 89777948 IC50 = 64 nM T70977 C1OV9A 89777949 IC50 = 26 nM T70977 C6KF0W 89777950 IC50 = 560 nM T70977 CQ7A9I 89777976 IC50 = 530 nM T70977 CR25EK 90353037 IC50 = 3180 nM T70977 C13KHM 90353051 IC50 = 7780 nM T70977 CF23HQ 90353109 IC50 = 2480 nM T70977 C7N5CP 90353119 IC50 = 7110 nM T70977 C3KWZ5 90488753 IC50 = 40000 nM T70977 C1WXC7 90644401 IC50 > 100000 nM T70977 CJ53FY 90644403 IC50 > 100000 nM T70977 CGUA74 90644405 IC50 > 100000 nM T70977 CW9Z3N 90644407 IC50 > 100000 nM T70977 CT27SY 90644409 IC50 > 100000 nM T70977 CMB4Q1 90644410 IC50 > 100000 nM T70977 CF0ZS7 90644412 IC50 > 100000 nM T70977 C1CM0J 90644414 IC50 > 100000 nM T70977 CS1Y2A 90644416 IC50 > 100000 nM T70977 CKJ16V 90644418 IC50 > 100000 nM T70977 CKH45I 90644420 IC50 > 100000 nM T70977 C3XTN6 90644422 IC50 > 100000 nM T70977 CEHV08 90644424 IC50 > 100000 nM T70977 CCR32H 90644426 IC50 > 100000 nM T70977 CA32ED 90644428 IC50 > 100000 nM T70977 CDS9Y8 90644430 IC50 > 100000 nM T70977 CEPL28 90644432 IC50 > 100000 nM T70977 C56RMJ 90644434 IC50 > 100000 nM T70977 CFW89O 90644436 IC50 > 100000 nM T70977 CY3NH1 90644438 IC50 > 100000 nM T70977 CC9FY8 90644440 IC50 > 100000 nM T70977 CYV14P 90644442 IC50 > 100000 nM T70977 CY0UC4 90645194 IC50 > 10000 nM T70977 C26BSU 90666124 IC50 > 10000 nM T70977 CVQ1O6 90666126 IC50 > 10000 nM T70977 C5AN9J 90666128 IC50 > 10000 nM T70977 CP76NE 90666130 IC50 > 10000 nM T70977 C85GHD 90666131 IC50 > 10000 nM T70977 CRP9I5 90666132 IC50 > 10000 nM T70977 CQI74X 90667795 Ki = 5400 nM T70977 CU5X3Z 90667796 Ki > 1000000 nM T70977 C4LF5U 90667797 Ki = 9000 nM T70977 C57LNQ 90667799 Ki = 4400 nM T70977 CI34EF 90667800 Ki = 4800 nM T70977 CO1E7Q 91667413 IC50 = 74 nM T70977 CQU2N5 91667414 IC50 = 5.9 nM T70977 CCKR05 91885622 IC50 = 8000 nM T70977 C0Y8ZK 91933875 IC50 > 10 nM T70977 CJQ5N6 91936970 IC50 = 682000 nM T70977 CAU45T 91971978 IC50 > 30000 nM T70977 COM94X 117072455 IC50 = 3.4 nM T70977 C7V5KF 117761549 IC50 = 350 nM T70977 C0Q8ZS 117762724 IC50 = 560 nM T70977 C7XUO9 118450030 IC50 = 31010 nM T70977 CB56VQ 118577456 IC50 = 14670 nM T70977 CY7BI2 118706214 IC50 > 10000 nM T70977 CS79AR 118707111 IC50 = 240000 nM T70977 CVW1O6 118707115 IC50 = 400000 nM T70977 CR4Z8V 118707118 IC50 = 750000 nM T70977 C3YAN0 118723092 IC50 = 10000 nM T70977 CR2Z4E 118727270 IC50 = 154.1 nM T70977 CBF5J3 118727271 IC50 = 105.4 nM T70977 CFV2M1 118727272 IC50 = 188 nM T70977 CUR8M9 118727273 IC50 = 204.1 nM T70977 CLX13T 118727274 IC50 = 74.1 nM T70977 C4FD3E 118727275 IC50 = 159.3 nM T70977 CY8U9Z 118727276 IC50 = 63.5 nM T70977 C1WL5K 118727277 IC50 = 327.4 nM T70977 C0GXT5 118727278 IC50 = 941.8 nM T70977 C0K1IV 118727279 IC50 = 73.6 nM T70977 CFYW70 118727280 IC50 = 69.7 nM T70977 CKF9M6 118727281 IC50 = 13 nM T70977 CULC92 118727282 IC50 = 36 nM T70977 C7T4XZ 118727283 IC50 = 120.6 nM T70977 CP5HR8 118727284 IC50 = 199.7 nM T70977 CCO91U 118732130 IC50 = 13 nM T70977 C32NSP 118732131 IC50 = 37 nM T70977 CI62CS 118732132 IC50 = 0.45 nM T70977 CMU40Y 118732133 IC50 = 0.29 nM T70977 C2A3IN 118732134 IC50 = 0.37 nM T70977 CNG0F4 118732135 IC50 = 30 nM T70977 C67XAN 118732136 IC50 = 2.4 nM T70977 CL2B9F 118732137 IC50 = 11 nM T70977 C1HE6U 118732138 IC50 = 2.4 nM T70977 C2ZF6Q 118732139 IC50 = 4.7 nM T70977 C49ULI 118732140 IC50 = 730 nM T70977 C3H7FJ 118732141 IC50 = 240 nM T70977 C2Y7CS 118732142 IC50 = 7.5 nM T70977 CVPS72 118732143 IC50 = 610 nM T70977 C9FOJ7 118732144 IC50 = 90 nM T70977 CY2RP1 118732145 IC50 = 7 nM T70977 C8XR4W 118732146 IC50 = 22 nM T70977 C2D4IR 118732147 IC50 = 6.8 nM T70977 CPW65L 118732148 IC50 = 4.4 nM T70977 CVEF32 118732149 IC50 = 24 nM T70977 C1DYA9 118732150 IC50 = 30 nM T70977 C84PGC 118732151 IC50 = 0.83 nM T70977 CK8U9A 118732152 IC50 = 140 nM T70977 CQCX41 118737057 IC50 > 10000 nM T70977 C42GSX 122180520 Ki > 4000 nM T70977 C4X7SD 122192466 IC50 > 10000 nM T70977 C32YBQ 122194770 IC50 = 140 nM T70977 CQ63PD 127025624 IC50 = 5560 nM T70977 C7M2LI 127025625 IC50 = 9060 nM T70977 CJT62C 127025626 IC50 = 9660 nM T70977 CY53OH 127027133 IC50 = 900 nM T70977 CMB8H5 127027134 IC50 = 2090 nM T70977 CDG0C4 127027135 IC50 = 2780 nM T70977 C6N0XM 127027136 IC50 = 2010 nM T70977 CN50FI 127027450 IC50 = 2490 nM T70977 C0Q7EF 127027451 IC50 = 9630 nM T70977 CTB46J 127027772 IC50 = 8300 nM T70977 C8TQ2G 127027773 IC50 = 12810 nM T70977 CBQ4E1 127027774 IC50 = 16990 nM T70977 CS4PK2 127034979 IC50 = 510 nM T70977 CQY49X 127035080 IC50 = 45 nM T70977 CCK32H 127035418 IC50 = 1200 nM T70977 CG43PQ 127035595 IC50 = 1000 nM T70977 CF1R5V 127035596 IC50 = 1700 nM T70977 CTOF48 127036309 IC50 = 210 nM T70977 C4XDZ1 127037287 IC50 = 112 nM T70977 CRX25F 127037288 IC50 = 67 nM T70977 C5Z7RP 127037289 IC50 = 39 nM T70977 CFST89 127037292 IC50 = 20 nM T70977 C0UZ4G 127037293 IC50 = 40 nM T70977 COGB08 127039586 IC50 = 100000 nM T70977 C63NOR 127039929 IC50 > 100000 nM T70977 C8DC4R 127040286 IC50 = 600 nM T70977 C52XTK 127044458 IC50 = 190 nM T70977 CG7ZQ4 127044481 IC50 = 135 nM T70977 C3TP9O 127044482 IC50 = 157 nM T70977 CBR56K 127044640 IC50 = 561 nM T70977 C8S0MO 127044806 IC50 = 184 nM T70977 CS5UM3 127044811 IC50 = 379 nM T70977 CV1E4O 127044959 IC50 = 157 nM T70977 C3S0NX 127044960 IC50 = 145 nM T70977 CT28ME 127044961 IC50 = 122 nM T70977 CGY19R 127044962 IC50 = 134 nM T70977 CM0YH9 127044963 IC50 = 173 nM T70977 CYS8P5 127044964 IC50 = 76 nM T70977 C54BUT 127044965 IC50 = 151 nM T70977 CMUF38 127044966 IC50 = 107 nM T70977 CF4N2W 127044967 IC50 = 406 nM T70977 CNOZ39 127044968 IC50 = 582 nM T70977 CT03ZN 127044969 IC50 = 92 nM T70977 COP85N 127044974 IC50 = 205 nM T70977 COS6B2 127044975 IC50 = 148 nM T70977 C83IXE 127044976 IC50 = 124 nM T70977 C7T8KX 127044977 IC50 = 80 nM T70977 C5X6AD 127044978 IC50 = 105 nM T70977 CP1A9T 127044979 IC50 = 72 nM T70977 C0PW1Y 127045571 IC50 = 293 nM T70977 C2LWZ1 129318964 IC50 = 1594 nM T70977 CUO41K 130470684 IC50 > 100000 nM T70977 CZ2JQ4 132427688 IC50 = 66 nM T70977 C4Q5LF 132471857 IC50 = 260 nM T70977 CB12WF 132575131 IC50 = 178000 nM T70977 C4EB8Y 134132531 IC50 > 50000 nM T70977 CFN34A 134132562 IC50 = 1450 nM T70977 CF6IK4 134135973 IC50 = 752 nM T70977 C7P2BG 134136529 IC50 = 45.7 nM T70977 CE69CG 134138526 IC50 = 180 nM T70977 CJZ9O3 134138839 IC50 = 43.5 nM T70977 CN7FR6 134140139 IC50 = 32 nM T70977 C9R1XV 134143185 IC50 > 50000 nM T70977 C8D7QS 134143690 IC50 = 1030 nM T70977 C6UEI4 134145833 IC50 = 356 nM T70977 CXI8Y1 134148934 IC50 > 50000 nM T70977 C4A0EG 134149314 IC50 = 19 nM T70977 CP3R1M 134152232 IC50 = 2610 nM T70977 CH0KU2 134153321 IC50 = 15700 nM T70977 C8FYC6 134153953 IC50 = 18000 nM T70977 C8N7BC 134154950 IC50 = 49 nM T70977 CUO21C 134156088 IC50 = 248 nM T70977 CU6FJ7 134157982 IC50 = 322000 nM T70977 C2AN7T 134611886 IC50 > 100000 nM T70977 CX0UR7 134694318 IC50 > 100000 nM T70977 C6X4LW 134816069 Ki = 70 nM T70977 CK7RY6 134816070 Ki = 9 nM T70977 CSZM60 134816433 Ki > 4000 nM T70977 CNK2R8 134816533 Ki = 190 nM T70977 C54FXD 134957362 IC50 > 10000 nM T70977 C8S0OH 135416016 IC50 = 24 nM T70977 C3YPB0 135416046 IC50 = 4 nM T70977 CMCS05 135420896 IC50 = 21000 nM T70977 CUL80S 135421123 IC50 = 4 nM T70977 CH23EZ 135432193 IC50 = 3000 nM T70977 CJZU04 135433406 IC50 = 1200 nM T70977 CHZ03C 135433925 IC50 = 55 nM T70977 CS6AM7 135434951 IC50 = 6500 nM T70977 CHM10I 135434952 IC50 = 520 nM T70977 CYH9W1 135434953 IC50 = 1800 nM T70977 CM75VI 135434962 IC50 = 3.981 nM T70977 C52RQG 135435008 IC50 = 8 nM T70977 CBN98A 135435009 IC50 = 8 nM T70977 CN6HJ9 135435010 IC50 = 36 nM T70977 CPFI68 135435011 IC50 = 0.8 nM T70977 C97ABO 135435012 IC50 = 1 nM T70977 CPXC89 135435013 IC50 = 6 nM T70977 CIX53V 135435014 IC50 = 12 nM T70977 CNM94K 135435015 IC50 = 1 nM T70977 CS14KX 135435016 IC50 = 5 nM T70977 C2ICP3 135435017 IC50 = 7 nM T70977 C6AZ2R 135435018 IC50 = 15 nM T70977 CTP7V8 135435022 IC50 > 10000 nM T70977 CN8M2G 135435823 IC50 = 27.7 nM T70977 CDU7X8 135438973 IC50 = 710 nM T70977 CJ7S0L 135444626 Ki < 2 nM T70977 CXP3N5 135453289 IC50 = 3000 nM T70977 CU96TX 135469872 IC50 > 10000 nM T70977 C09BEG 135486057 IC50 > 10000 nM T70977 CUJ86P 135494240 IC50 = 500 nM T70977 CU97NR 135510708 IC50 = 110 nM T70977 CL5IR0 135512024 IC50 = 80 nM T70977 C0XV8S 135512471 IC50 = 1800 nM T70977 C6B9TE 135514366 IC50 = 6080 nM T70977 C4NV7G 135518519 IC50 = 40 nM T70977 CTJ48K 135524085 IC50 = 530 nM T70977 CUT1W7 135524168 IC50 = 300 nM T70977 CS57UE 135533150 IC50 = 18030 nM T70977 C8T1KE 135537879 IC50 > 10000 nM T70977 CKF13W 135546072 IC50 = 5000 nM T70977 C5API7 135558907 IC50 = 100 nM T70977 CTB7R2 135564980 IC50 = 7700 nM T70977 CRD8M3 135566516 IC50 = 55000 nM T70977 C0BHA5 135574941 IC50 = 27.1 nM T70977 CCO3K7 135580426 IC50 = 5.012 nM T70977 CMR62I 135583974 IC50 = 0.7 nM T70977 CPV59N 135685787 Ki = 2 nM T70977 C4Y2CG 135686834 Ki = 99 nM T70977 CG9R0V 135741827 IC50 > 10000 nM T70977 CCB75F 135753920 IC50 = 2400 nM T70977 C3WR5H 135753941 IC50 = 1300 nM T70977 CHX05K 135753962 IC50 = 1300 nM T70977 CGPI93 135753969 IC50 = 2100 nM T70977 CUFI29 135753973 IC50 = 8900 nM T70977 CU7Q6H 135778711 IC50 > 10000 nM T70977 CC76HV 135778712 IC50 > 10000 nM T70977 CY4UO9 135778713 IC50 = 3162.28 nM T70977 CSU89F 135778714 IC50 = 2511.89 nM T70977 C5LFC6 135778715 IC50 > 10000 nM T70977 COR9P4 135778716 IC50 = 12.59 nM T70977 CNOF40 135848025 IC50 = 27 nM T70977 CF6AK5 135848026 IC50 = 149000 nM T70977 CY7ZQ6 135848030 IC50 = 98000 nM T70977 CZ8VL4 135848031 IC50 = 49000 nM T70977 C5L0XB 135848037 IC50 = 56000 nM T70977 CBJ85I 135848038 IC50 = 14000 nM T70977 CZ5D0P 135853872 IC50 = 3960 nM T70977 CMW9G4 135897727 IC50 = 128.82 nM T70977 C02PHA 135927892 IC50 = 630.96 nM T70977 CS8T3D 135927897 IC50 = 1584.89 nM T70977 CF1PS8 135934877 Ki = 0.8 nM T70977 C6H0AI 135957039 IC50 = 6760 nM T70977 CX79TY 135957045 IC50 = 100 nM T70977 CGI8Y6 135957348 IC50 = 4160 nM T70977 C7J9SG 135965869 IC50 = 39 nM T70977 CQ3NP8 135976588 Ki = 8.3 nM T70977 C26ASG 135976589 Ki = 23 nM T70977 C65QDA 135976590 Ki = 16 nM T70977 CBG36C 135976591 Ki = 7.7 nM T70977 C0A7PZ 135976592 Ki = 50 nM T70977 CEN58K 135976613 Ki > 3700 nM T70977 CJ5A1Q 135976614 Ki = 650 nM T70977 C4VT8B 135976615 Ki = 200 nM T70977 C5KL2Y 135976616 Ki = 250 nM T70977 C5AJI0 135976617 Ki = 720 nM T70977 C9NTA4 135976618 Ki = 850 nM T70977 C2A8MT 135976619 Ki = 44 nM T70977 CCAO27 135976620 Ki = 120 nM T70977 CI5TS0 135976621 Ki > 4000 nM T70977 CS75RO 135976622 Ki = 35 nM T70977 C2DAY9 135976623 Ki = 20 nM T70977 C6B5RL 135976624 Ki = 640 nM T70977 CIA08P 135976625 Ki = 20 nM T70977 CH6G7M 135976626 Ki = 30 nM T70977 CFXG69 135976627 Ki = 18 nM T70977 CX1Q5O 135976628 Ki = 2 nM T70977 CM76AP 135976629 Ki < 2 nM T70977 CF38CU 135976630 Ki = 9 nM T70977 C1JBC6 135976631 Ki = 2 nM T70977 CK5MC9 135976632 Ki = 39 nM T70977 C19PHF 135976633 Ki = 8 nM T70977 CGSZ58 135976634 Ki = 9 nM T70977 C3LN0J 135976635 Ki = 5 nM T70977 C0UXE3 135976636 Ki = 4 nM T70977 CSP6L3 135976637 Ki = 8 nM T70977 C2PS3K 135976638 Ki = 30 nM T70977 CNPR50 135976639 Ki = 23 nM T70977 C0KWS6 135976640 Ki = 6.5 nM T70977 CV3QM7 135976641 Ki = 9 nM T70977 C0N5GY 135976642 Ki = 59 nM T70977 CUAX40 135976643 Ki = 1.9 nM T70977 CNYC46 135976644 Ki = 2 nM T70977 C2UM0Z 135976645 Ki < 2 nM T70977 CD80SR 135976646 Ki = 14 nM T70977 CG2YO7 135976647 Ki = 110 nM T70977 CY13GJ 135976648 Ki = 16 nM T70977 CX0TK9 135976650 Ki = 8 nM T70977 CY2L8G 135976651 Ki < 3.5 nM T70977 C7W3GS 135976652 Ki = 0.4 nM T70977 C1SFB3 135976653 Ki = 0.4 nM T70977 CPM95Y 135976654 Ki < 2 nM T70977 CRLZ83 135976655 Ki < 3.5 nM T70977 CY0C5A 135976656 Ki < 3.5 nM T70977 C7MN5V 135976657 Ki = 87 nM T70977 C83ULT 135976658 Ki = 2 nM T70977 C0XU7A 135976659 Ki = 3 nM T70977 CTRL59 135976660 Ki = 4.5 nM T70977 CWX7Y9 135976661 Ki = 3 nM T70977 C2RV9I 135976662 Ki = 270 nM T70977 CKF69A 135976663 Ki = 3.7 nM T70977 CXH30P 135978796 IC50 = 1.5 nM T70977 CNI6A4 135996019 IC50 = 477.2 nM T70977 C8EPO5 135998745 IC50 > 1000 nM T70977 CHA4N2 136013680 IC50 > 10 nM T70977 CDA5Q0 136016378 IC50 = 100 nM T70977 CBS87V 136016385 IC50 = 540 nM T70977 C05IWG 136016386 IC50 = 1260 nM T70977 COPL16 136016393 IC50 = 2290 nM T70977 C8T5ZB 136016456 IC50 = 5900 nM T70977 CFT3I1 136026170 IC50 = 90 nM T70977 CKG9Z4 136040144 IC50 = 40180 nM T70977 CE43UZ 136041855 IC50 > 1000 nM T70977 C79XQW 136042384 IC50 = 110 nM T70977 CFS02H 136059694 IC50 = 5 nM T70977 C4B8AI 136123466 IC50 = 160 nM T70977 CC6PG2 136174827 IC50 = 6030 nM T70977 CMP8X1 136188793 IC50 = 2400 nM T70977 C1YUD0 136219394 IC50 > 10 nM T70977 C6EY3K 136223992 IC50 = 5 nM T70977 C5RI6D 136224254 IC50 > 10000 nM T70977 CT9VC6 136224366 IC50 > 10000 nM T70977 CF6B3S 136224367 IC50 > 10000 nM T70977 C4OQ1U 136240234 IC50 < 50000000 nM T70977 C83OBX 136241622 IC50 = 830 nM T70977 C80OEU 136245075 IC50 = 7310 nM T70977 C6S1GT 136245126 IC50 > 10000 nM T70977 CS6K0B 136245127 IC50 > 10000 nM T70977 CA5KP8 136245128 IC50 > 10000 nM T70977 CRTI72 136249339 IC50 = 2.5 nM T70977 CY36QB 136254272 IC50 = 250 nM T70977 CIU8W3 136254389 IC50 > 10 nM T70977 C8UQ7C 136264319 IC50 > 10000 nM T70977 CNE6I8 136264499 IC50 > 10000 nM T70977 CL95WA 136380901 IC50 = 6.1 nM T70977 CRB3M4 136609929 IC50 > 10000 nM T70977 C0A9VE 136609930 IC50 > 10000 nM T70977 CW5YL0 136609931 IC50 > 10000 nM T70977 C7EAJ9 136980453 IC50 = 515 nM T70977 CL1EB7 137283359 IC50 = 44.3 nM T70977 C3R5AW 137287456 IC50 = 24 nM T70977 CL38VG 137287457 IC50 = 2.1 nM T70977 CGAN83 137287458 IC50 = 51.7 nM T70977 CNFE23 137349058 IC50 = 80 nM T70977 CV6KR8 137349062 IC50 = 250 nM T70977 C8DF0S 137349068 IC50 = 2 nM T70977 CURM83 137349070 IC50 = 430 nM T70977 CM26KA 137628998 IC50 = 510 nM T70977 CBDU81 137629200 IC50 = 14 nM T70977 C6R2PY 137630916 IC50 = 1895 nM T70977 CK5WC1 137632241 IC50 = 13860 nM T70977 C4GK6S 137632595 IC50 = 1.8 nM T70977 CVL41R 137633869 IC50 = 1010 nM T70977 CS4D2Q 137634160 IC50 = 11 nM T70977 CI1E8V 137634241 IC50 > 10000 nM T70977 CC3J8N 137635045 IC50 > 20000 nM T70977 C5CRX4 137635152 IC50 = 12 nM T70977 C8GQD5 137636872 IC50 = 91 nM T70977 CW9K4H 137636941 IC50 = 660 nM T70977 CR9IZ6 137637770 IC50 = 11 nM T70977 CT8PZ0 137638234 IC50 = 1.7 nM T70977 C1KP0C 137639235 IC50 = 1200 nM T70977 C4XEI1 137639320 IC50 = 5160 nM T70977 CR3AV7 137639578 IC50 > 20000 nM T70977 CKHD52 137639853 IC50 = 22 nM T70977 C7PNM9 137640981 IC50 > 20000 nM T70977 CC37FW 137641147 IC50 = 3000 nM T70977 C7TG3J 137641313 IC50 = 457.09 nM T70977 C2VOW8 137641402 IC50 = 7.4 nM T70977 CET86D 137641554 IC50 > 20000 nM T70977 CI17FX 137641801 IC50 = 15290 nM T70977 CH21YK 137642640 IC50 = 1.8 nM T70977 CUB38E 137642944 IC50 = 0.9 nM T70977 CAKC72 137642992 IC50 = 20 nM T70977 C2CHB5 137643012 IC50 = 2 nM T70977 CZL28M 137643099 IC50 = 24 nM T70977 C4DRX1 137643187 IC50 = 5300 nM T70977 CA2SO9 137644063 IC50 > 10000 nM T70977 C74DEQ 137644716 IC50 = 15840 nM T70977 CDA2N6 137644922 IC50 = 51 nM T70977 CM2DS6 137645628 IC50 = 0.73 nM T70977 CH9DO7 137646393 IC50 = 8.2 nM T70977 CN4S1M 137646665 IC50 = 8.1 nM T70977 C0M6DZ 137647193 IC50 = 56 nM T70977 COW27K 137647779 IC50 = 9230 nM T70977 C7B3SG 137649023 IC50 = 25 nM T70977 C91HPM 137649287 IC50 = 26 nM T70977 CDJ65E 137649524 IC50 = 26 nM T70977 CLE6S3 137649674 IC50 = 111 nM T70977 CMG94F 137649707 IC50 = 110 nM T70977 C7PMO3 137650008 IC50 = 5 nM T70977 CP9EN8 137650185 IC50 = 9610 nM T70977 CW04TZ 137650486 IC50 = 4780 nM T70977 CT36PX 137650758 IC50 = 220 nM T70977 C3LG5H 137650873 IC50 = 15 nM T70977 C9DI5N 137650897 IC50 = 11 nM T70977 CL7ZX9 137651411 IC50 = 0.25 nM T70977 C6GJA5 137651722 IC50 = 4.7 nM T70977 CY54EU 137654374 IC50 = 3.5 nM T70977 C1U5PD 137654853 IC50 = 3000 nM T70977 C8TDA4 137655242 IC50 = 7580 nM T70977 C20ALD 137655637 IC50 > 20000 nM T70977 CGW9I0 137656387 IC50 = 5010 nM T70977 CY32TC 137657744 IC50 = 18 nM T70977 C5JF2T 137658198 IC50 = 1.2 nM T70977 CC34LO 137658348 IC50 = 1140 nM T70977 C3TY9U 137658647 IC50 = 810 nM T70977 CZB26I 137658958 IC50 > 20000 nM T70977 CI7FU6 137659802 IC50 = 7500 nM T70977 CD9W1H 137660657 IC50 = 12700 nM T70977 C3B6MD 137661138 IC50 = 2 nM T70977 CEI0F4 137661223 IC50 = 290 nM T70977 C79JRM 137661247 IC50 > 10000 nM T70977 CP63IC 137661560 IC50 = 6.7 nM T70977 CIW2G0 137662322 IC50 = 22 nM T70977 CA3G0W 140534484 IC50 = 308 nM T70977 CGUA35 142598857 IC50 > 10000 nM T70977 CLO0R1 142737566 IC50 = 33800 nM T70977 C0WXF6 142737574 IC50 > 50000 nM T70977 CHI9R4 142737576 IC50 = 994 nM T70977 CCNU56 142737578 IC50 = 1.37 nM T70977 C6VB3O 145925651 IC50 >= 5000 nM T70977 CC85FJ 145949364 IC50 = 9220 nM T70977 CBCS01 145949465 IC50 = 2 nM T70977 CEI51C 145951560 IC50 > 10000 nM T70977 CFN52Q 145952674 IC50 = 7470 nM T70977 C1W0GJ 145952796 IC50 = 31622.78 nM T70977 C2YF6H 145953038 IC50 = 1.6 nM T70977 C2V6FM 145955631 IC50 = 1.1 nM T70977 CHJ8I4 145956228 IC50 = 3550 nM T70977 CJF9A4 145956684 IC50 = 890 nM T70977 CFR51Q 145957334 IC50 = 1.3 nM T70977 C3MTG8 145957448 IC50 = 5.2 nM T70977 CZG32V 145958978 IC50 = 1.3 nM T70977 CNG5O7 145960049 IC50 = 8540 nM T70977 CZO6T7 145961089 IC50 > 25118.86 nM T70977 CX6T3J 145961172 IC50 = 2511.89 nM T70977 C54ZQA 145961234 IC50 > 25118.86 nM T70977 C83FPK 145961240 IC50 = 31.62 nM T70977 C31QBE 145961348 IC50 > 25118.86 nM T70977 COCG81 145961565 IC50 = 7943.28 nM T70977 C73MVW 145961583 IC50 = 15848.93 nM T70977 C6HB9M 145961899 IC50 = 19952.62 nM T70977 CLFQ85 145963006 IC50 = 398.11 nM T70977 CYZ14S 145963250 IC50 > 25118.86 nM T70977 CAD5Q9 145963302 IC50 > 25118.86 nM T70977 C35ZRP 145963416 IC50 = 7943.28 nM T70977 C3VQN6 145964437 IC50 = 50000 nM T70977 CB32OW 145964815 IC50 > 50000 nM T70977 CVG34Q 145965154 IC50 > 50000 nM T70977 C6HD7A 145966030 IC50 = 8100 nM T70977 C3ITW7 145966076 IC50 = 6900 nM T70977 C4OEW5 145966583 IC50 > 50000 nM T70977 C1L4BR 145966694 IC50 > 50000 nM T70977 CDNC31 145967951 IC50 > 500 nM T70977 C82GAM 145972125 Ki = 6300 nM T70977 CV0L6A 145972558 IC50 = 50000 nM T70977 C35LOD 145973081 IC50 = 25600 nM T70977 CTW56H 145973391 IC50 = 280 nM T70977 CI1S0B 145973974 IC50 > 50000 nM T70977 CZE89S 145974229 IC50 = 10100 nM T70977 CGB7L4 145974437 IC50 = 5400 nM T70977 CISH58 145975235 IC50 = 2350 nM T70977 C43GFI 145975558 IC50 = 10000 nM T70977 C0KXH4 145975825 IC50 = 50000 nM T70977 CTFJ90 145975836 IC50 = 8100 nM T70977 C40HMI 145976797 IC50 = 4100 nM T70977 CMZ81R 145976977 IC50 = 8700 nM T70977 C31FEQ 145977262 IC50 > 50000 nM T70977 CD5KI4 145977612 IC50 = 21200 nM T70977 CQ7DM1 145977815 IC50 > 50000 nM T70977 CZ6K5O 145978604 IC50 > 50000 nM T70977 CS5FJ3 145979187 IC50 = 17000 nM T70977 CC9FX6 145979710 IC50 = 28000 nM T70977 C38KWC 145979876 IC50 = 35000 nM T70977 CTA95I 145979993 IC50 = 18000 nM T70977 CIR5M6 145980012 IC50 = 670 nM T70977 CGDP36 145980029 IC50 = 65 nM T70977 C78GKB 145980118 IC50 = 75000 nM T70977 C69EZH 145980213 IC50 = 22000 nM T70977 C23KST 145980531 IC50 = 90000 nM T70977 CO9F3K 145981169 IC50 = 20000 nM T70977 CT02VJ 145981438 IC50 = 11400 nM T70977 CU1RE3 145981895 IC50 = 6000 nM T70977 C8RN0E 145982001 IC50 = 63 nM T70977 CLD9H6 145982286 IC50 = 99 nM T70977 CROC78 145983700 IC50 = 51000 nM T70977 CG83SB 145984620 IC50 = 25000 nM T70977 C38JVG 145984879 IC50 = 49000 nM T70977 C19IWK 145986527 IC50 = 270 nM T70977 CV5GN1 145986655 IC50 = 27000 nM T70977 CGDM47 145987297 IC50 = 35000 nM T70977 C6CAP4 145987452 IC50 = 19000 nM T70977 CXF27U 145987502 IC50 = 45000 nM T70977 CK5M9W 145987607 IC50 = 2500 nM T70977 CJP7H5 145987783 IC50 = 18 nM T70977 C6Y8LK 145988014 IC50 = 80000 nM T70977 CJ4U7L 145988121 IC50 = 98 nM T70977 CD7K3H 145988440 IC50 = 13600 nM T70977 CCE2Y3 145988467 IC50 = 18000 nM T70977 C79RBC 145989455 IC50 = 35000 nM T70977 CN6C4X 145990029 IC50 = 5300 nM T70977 CRSD39 145990133 IC50 > 100000 nM T70977 CD6P8X 145990469 IC50 = 27000 nM T70977 CW5H3N 145990758 IC50 = 1500 nM T70977 CI6JL2 145990903 IC50 = 48000 nM T70977 CPSB67 145991106 IC50 = 33000 nM T70977 CZTM79 145991359 IC50 = 20000 nM T70977 CBH98M 145991372 IC50 = 21000 nM T70977 C2JO1W 145991711 IC50 > 100000 nM T70977 C8KUE6 145991747 IC50 = 180 nM T70977 CPJ26A 145991919 IC50 = 18000 nM T70977 CR69KG 145992024 IC50 = 68 nM T70977 C19GZS 145992418 IC50 = 83 nM T70977 CF4NY0 145992429 IC50 = 66000 nM T70977 CLF28N 145992533 IC50 = 4600 nM T70977 C1FBD7 145993205 IC50 = 34 nM T70977 CQR8U6 145993560 IC50 = 100000 nM T70977 C94AOS 145993818 IC50 = 25000 nM T70977 CT5Y2D 145993819 IC50 = 32000 nM T70977 CZ06PL 149855821 IC50 > 10000 nM T70977 CY5H6I 151422375 IC50 = 315 nM T70977 C7K8BU 151918601 IC50 = 891 nM T70977 CEX76V 152449061 IC50 = 1204 nM T70977 C4K8TH 154777683 IC50 = 767 nM T70977 CUP08F 154778142 IC50 = 565 nM T70977 CRAD72 154778144 IC50 = 1196 nM T70977 CUH9P6 155077159 IC50 = 108.4 nM T70977 CV0MZ9 155510817 IC50 = 215 nM T70977 CXWI87 155511357 IC50 > 10000 nM T70977 CO5WR4 155511447 IC50 = 170 nM T70977 CD8M7Q 155512392 IC50 = 663 nM T70977 CG3TS5 155512736 IC50 > 10000 nM T70977 C2MD1Q 155513187 IC50 > 10000 nM T70977 C2D6UL 155513283 IC50 > 10000 nM T70977 CD0SG7 155514146 IC50 = 354 nM T70977 COM30P 155514391 Ki = 650 nM T70977 C6SQX5 155514684 IC50 = 527 nM T70977 CP4UQ3 155515929 IC50 = 808 nM T70977 CF3CZ6 155516064 IC50 = 3760 nM T70977 CS5ZQ1 155516197 IC50 = 629 nM T70977 CL47DJ 155516579 IC50 = 19960 nM T70977 CR6D8T 155516775 IC50 = 22.8 nM T70977 CL7G5U 155517186 IC50 = 4110 nM T70977 C12DHX 155517839 IC50 = 13 nM T70977 CR1A0B 155518258 IC50 = 739 nM T70977 C7U0CL 155519223 IC50 = 86 nM T70977 C4P1RM 155520291 IC50 = 2690 nM T70977 C0NMJ7 155520623 IC50 = 428 nM T70977 C83RWF 155520850 IC50 = 2.75 nM T70977 C86ALD 155521765 IC50 = 1499 nM T70977 CPX8J2 155521813 IC50 = 62.1 nM T70977 CIK2W8 155522314 IC50 = 91 nM T70977 CL62FA 155522342 IC50 = 232.9 nM T70977 CC56HQ 155522585 IC50 > 10000 nM T70977 CHF31J 155522721 IC50 = 893 nM T70977 C3HE8T 155522847 IC50 > 2000 nM T70977 C9KU0T 155523035 IC50 = 2260 nM T70977 CDJH54 155523269 IC50 = 260 nM T70977 CQW9M3 155523312 IC50 = 1149 nM T70977 C9NM7B 155523411 IC50 = 39 nM T70977 C9WH1A 155523541 IC50 = 38 nM T70977 CCTW17 155524059 IC50 = 4343 nM T70977 CV8P9Q 155524146 IC50 > 10000 nM T70977 C76ZQG 155524866 IC50 = 110 nM T70977 C0T3AK 155524940 IC50 = 418 nM T70977 CW3S9D 155525178 IC50 = 53 nM T70977 CW96RL 155525249 IC50 = 47 nM T70977 CEIW40 155525530 IC50 = 117 nM T70977 C0S7GV 155525697 IC50 > 10000 nM T70977 C4F9QH 155525702 IC50 = 265 nM T70977 C9HKF7 155526015 IC50 = 64 nM T70977 C78LEV 155526363 IC50 = 372 nM T70977 C5H1UB 155526385 IC50 = 1758 nM T70977 CCGD64 155526869 IC50 = 183 nM T70977 C9BMN4 155527815 IC50 = 1252 nM T70977 CLT3E4 155527966 IC50 = 99 nM T70977 C2MI4C 155528595 IC50 > 10000 nM T70977 CEXY67 155528636 IC50 = 79 nM T70977 C2OVI6 155529891 IC50 = 3.59 nM T70977 CE5WL9 155530746 IC50 = 20000 nM T70977 C8FER3 155531005 IC50 > 10000 nM T70977 C0QO5E 155531724 IC50 = 72 nM T70977 COU0M7 155532838 IC50 = 71 nM T70977 C0C2OE 155533282 IC50 = 0.508 nM T70977 CBNX32 155535545 IC50 = 127 nM T70977 CK6N2W 155535911 IC50 = 167 nM T70977 C6UDV1 155536548 IC50 = 133 nM T70977 C7MS0B 155536931 IC50 = 155.4 nM T70977 C2CG1A 155537016 IC50 > 10000 nM T70977 CFC3D2 155537268 IC50 = 59 nM T70977 C9TXU8 155537377 IC50 = 23 nM T70977 C3ZHC0 155537470 IC50 = 18.46 nM T70977 C2A9KV 155537532 IC50 > 10000 nM T70977 CD4G8Y 155538105 IC50 = 4640 nM T70977 COE67I 155538620 IC50 = 59 nM T70977 CEP37L 155538694 IC50 = 156 nM T70977 CZD76V 155538756 IC50 > 10000 nM T70977 CS4W6B 155538942 IC50 = 510 nM T70977 COY2K6 155539289 IC50 = 347.9 nM T70977 C9UZJ6 155539371 IC50 = 43 nM T70977 CC0AJ1 155539740 IC50 = 148 nM T70977 C4LAT3 155539976 IC50 = 3 nM T70977 C87MOT 155540289 IC50 > 10000 nM T70977 C4ZT7J 155540573 IC50 = 1820 nM T70977 C5ORP4 155540981 IC50 = 4420 nM T70977 CBM39S 155541324 IC50 = 467 nM T70977 C32CFS 155541434 IC50 = 899 nM T70977 C8K3WL 155541562 IC50 = 956 nM T70977 C5IS0W 155541608 IC50 = 128 nM T70977 CDM03I 155541927 IC50 = 1429 nM T70977 C3J8SM 155542090 IC50 = 363 nM T70977 C9O1UR 155542967 IC50 = 77.1 nM T70977 C4KMP8 155543427 IC50 = 132 nM T70977 CQMZ76 155544092 IC50 = 3 nM T70977 C7YK0H 155544525 IC50 = 16.5 nM T70977 C8QF6I 155545556 IC50 = 1717 nM T70977 C15KRU 155545689 IC50 = 352 nM T70977 CHCS54 155546044 Ki = 530 nM T70977 CA1EJ5 155547420 IC50 = 770 nM T70977 C52SXT 155547535 IC50 = 199 nM T70977 COG6I5 155548241 IC50 = 571 nM T70977 CI4O2U 155548411 IC50 > 10000 nM T70977 CC52UD 155550429 IC50 = 240 nM T70977 C8PA6D 155550766 IC50 = 126 nM T70977 C36MZV 155551706 IC50 = 103 nM T70977 CEJ45N 155552201 IC50 = 130 nM T70977 CF9JS0 155552697 IC50 = 4.43 nM T70977 C9C4XO 155553435 IC50 = 229 nM T70977 CEBV41 155554010 IC50 = 542 nM T70977 C3I6NL 155554624 IC50 = 82 nM T70977 C95VTO 155554722 IC50 = 220 nM T70977 CV60MW 155555951 IC50 = 3654 nM T70977 CG4DT9 155556962 IC50 = 63.1 nM T70977 C9M4DG 155557125 IC50 = 3242 nM T70977 C4LY2S 155557392 IC50 = 2470 nM T70977 CVY7W6 155557769 IC50 = 49 nM T70977 CS8DI1 155558034 IC50 = 462 nM T70977 C92NTS 155558433 IC50 > 100000 nM T70977 C48FUJ 155558812 IC50 = 320 nM T70977 C5JRG0 155558848 IC50 = 11 nM T70977 CP18NC 155559676 IC50 = 47 nM T70977 CNX32F 155560561 IC50 = 570 nM T70977 CID3V4 155560946 IC50 = 4110 nM T70977 CJX20C 155561847 IC50 = 1684 nM T70977 C6D7OT 155562118 IC50 = 3090 nM T70977 CC2G3E 155562659 IC50 = 4210 nM T70977 CYGU28 155563030 IC50 = 4050 nM T70977 CRC25F 155563369 IC50 = 73 nM T70977 CPS4C6 155563814 IC50 = 5180 nM T70977 C31SXI 155563958 IC50 = 136 nM T70977 C16JFY 155563983 IC50 = 5460 nM T70977 C1DM5X 155564336 IC50 = 69 nM T70977 CS5FM6 155565596 IC50 = 219 nM T70977 CS9ZI1 155565616 IC50 = 1.42 nM T70977 C6OMA4 155565625 IC50 = 633 nM T70977 C8PY6V 155565896 IC50 = 64.2 nM T70977 CWGZ76 155566793 IC50 > 10000 nM T70977 CGX17T 155567824 IC50 = 236 nM T70977 CA7B0F 155568022 IC50 = 9850 nM T70977 CRD24F 155568639 IC50 = 560 nM T70977 C1S8ZB 155568922 IC50 = 550 nM T70977 CZBS25 155568984 IC50 = 471 nM T70977 CP06DW 155569342 IC50 = 576 nM T70977 D00AAN 23643731 IC50 = 7200 nM T70977 D00ERW 44444843 Ki > 7059 nM T70977 D00HUP 46894037 IC50 = 16 nM T70977 D00HVA 11624601 Ki > 7100 nM T70977 D00RIX 5280443 IC50 = 1900 nM T70977 D00SEC 3641059 IC50 = 920 nM T70977 D00TBD 10461815 IC50 > 10000 nM T70977 D00XUF 49863103 IC50 = 1220 nM T70977 D01IPF 22319573 IC50 = 94 nM T70977 D01MEP 6539732 IC50 = 390 nM T70977 D01OJG 6539451 IC50 = 520 nM T70977 D01RKI 23643732 IC50 = 23000 nM T70977 D02BIK 56603751 Ki = 2 nM T70977 D02DLC 6539361 Ki = 10 nM T70977 D02OPH 448008 IC50 = 76 nM T70977 D02QAZ 11612883 IC50 > 1000 nM T70977 D02XHC 448912 IC50 = 650 nM T70977 D02ZIY 10020713 IC50 = 5 nM T70977 D03DZO 11715767 IC50 = 220 nM T70977 D03OED 22319694 IC50 = 5008 nM T70977 D04ACJ 10380885 IC50 = 1353 nM T70977 D04PEI 11467730 IC50 = 36000 nM T70977 D04TPA 72163809 IC50 = 2600 nM T70977 D04VBD 10423871 IC50 = 198 nM T70977 D04ZWF 53396311 IC50 = 0.6 nM T70977 D05AMQ 6539137 IC50 = 70000 nM T70977 D05NKG 16760286 IC50 = 0.8 nM T70977 D05QML 16048421 IC50 = 35 nM T70977 D05SXF 25209788 IC50 = 53 nM T70977 D06HVH 54613583 IC50 > 10000 nM T70977 D06OAH 448949 IC50 = 174 nM T70977 D06YMZ 22319484 IC50 = 8525 nM T70977 D07ADX 54764565 IC50 > 10000 nM T70977 D07IVD 10266409 IC50 = 4140 nM T70977 D07OAT 456214 IC50 > 10000 nM T70977 D07OCA 5330812 IC50 = 210 nM T70977 D07PTD 10085013 IC50 = 390 nM T70977 D07WXT 433294 IC50 = 6530 nM T70977 D08HFG 24809764 IC50 = 1390 nM T70977 D09BQY 22319483 IC50 = 2459 nM T70977 D09FFE 449241 IC50 = 15000 nM T70977 D09HVH 135566652 IC50 > 10 nM T70977 D09VQM 442428 IC50 = 100000 nM T70977 D09ZNV 447682 IC50 = 14000 nM T70977 D0A1CM 5281855 IC50 = 7500 nM T70977 D0A1YQ 176158 IC50 = 7 nM T70977 D0A9MY 10085818 IC50 = 76 nM T70977 D0C9OT 10265187 IC50 = 195 nM T70977 D0CM6T 11314340 Ki = 110 nM T70977 D0D5ZL 369401 IC50 = 4 nM T70977 D0D6MH 11617559 IC50 > 32000 nM T70977 D0DR8N 6538897 IC50 = 18 nM T70977 D0E2XM 23643836 IC50 = 4800 nM T70977 D0E6GC 10085059 IC50 = 661 nM T70977 D0EU1R 46215815 IC50 > 25118 nM T70977 D0F0AX 135413546 IC50 = 10 nM T70977 D0F5EI 10017019 IC50 = 2000 nM T70977 D0G4GB 10757 IC50 = 50000 nM T70977 D0GN5Z 5281295 IC50 = 1950 nM T70977 D0H3EV 5005498 IC50 = 3.999 nM T70977 D0H4VB 71461150 IC50 = 53300 nM T70977 D0IL0G 9993220 IC50 = 260 nM T70977 D0J4ON 135473382 IC50 = 754 nM T70977 D0L0HG 766949 IC50 > 10000 nM T70977 D0L2WP 46225540 IC50 = 500 nM T70977 D0M3SC 22319511 IC50 = 14000 nM T70977 D0M5FF 5083 IC50 = 2.8 nM T70977 D0N4WB 4210951 Ki = 24 nM T70977 D0NL1F 23643835 IC50 = 5400 nM T70977 D0O0VP 6539367 Ki = 10 nM T70977 D0O6OH 71553154 IC50 = 7740 nM T70977 D0PT2D 9904289 IC50 = 1500 nM T70977 D0Q0YV 24944925 IC50 = 831.76 nM T70977 D0Q3KS 9957049 IC50 = 0.56 nM T70977 D0Q3NG 11715520 Ki > 7100 nM T70977 D0Q4QF 6509753 IC50 = 8400 nM T70977 D0Q7TO 6419766 Ki = 22 nM T70977 D0R5EF 10016510 IC50 = 5900 nM T70977 D0R5FH 438981 IC50 = 1000 nM T70977 D0R6TL 10421683 IC50 = 354 nM T70977 D0R7QL 23643537 IC50 = 10400 nM T70977 D0S3RP 135458003 IC50 = 44 nM T70977 D0S7IE 11658882 Ki > 7100 nM T70977 D0T1CE 22319580 IC50 = 935 nM T70977 D0T8KR 9549289 IC50 = 30 nM T70977 D0T8NU 16757525 IC50 = 146 nM T70977 D0TF9P 6538761 IC50 = 119.95 nM T70977 D0TO6S 2396 IC50 = 190.55 nM T70977 D0V6HG 46894038 IC50 = 26 nM T70977 D0X4CO 9847557 Ki = 0.09 nM T70977 D0Y0ES 3707 IC50 = 22 nM T70977 D0Y5RO 4566 IC50 = 40 nM T70977 D0YM4A 22319604 IC50 = 80 nM T70977 D0Z2CN 135418335 IC50 = 500 nM T99989 D0A3MV 448014 IC50 > 100000000 nM T99989 D0YK9D 9956119 IC50 > 5000 nM T99989 C5R1AG 2155128 IC50 = 4030 nM T99989 CF86YB 2155264 IC50 = 7070 nM T99989 CV86WR 2155389 IC50 > 10000 nM T99989 CPQV76 5353678 IC50 = 600 nM T99989 CY20RA 7458031 IC50 > 100000 nM T99989 C7T9ES 11681588 IC50 = 29 nM T99989 C1HO8W 18563036 IC50 = 7340 nM T99989 CJ76FL 22037373 IC50 = 305 nM T99989 CFMQ08 24370907 IC50 > 100000 nM T99989 CXZ84S 25143677 IC50 = 13.7 nM T99989 C2V5WQ 25143825 IC50 = 14.2 nM T99989 C7R8NQ 25143828 IC50 = 4.6 nM T99989 CKZ64S 25143829 IC50 = 14.6 nM T99989 C0EPV1 25143967 IC50 = 8.6 nM T99989 C9QMC5 25143969 IC50 = 43 nM T99989 C2U0NP 30291209 IC50 > 100000 nM T99989 C7S6OT 30291292 IC50 > 100000 nM T99989 C3VRO9 44557921 IC50 > 10000 nM T99989 C7D8ZN 44597226 IC50 = 73 nM T99989 C4HN5F 44597227 IC50 = 447 nM T99989 C6O7VL 53357600 IC50 = 28.2 nM T99989 C71OXL 53388145 IC50 = 15300000 nM T99989 CDL28G 53388146 IC50 > 100000000 nM T99989 CIM94L 56668847 IC50 > 100000000 nM T99989 C8PK0W 56675716 IC50 > 100000000 nM T99989 COTF12 57382553 IC50 = 27 nM T99989 CEW5L7 57522817 IC50 = 20000 nM T99989 C4SEH5 57522818 IC50 = 60000 nM T99989 CF8IP6 57522819 IC50 > 100000 nM T99989 CJ56CE 57522820 IC50 > 100000 nM T99989 C3XI2P 57523093 IC50 > 100000 nM T99989 CUH3B5 57523094 IC50 > 100000 nM T99989 C3QF2X 57523095 IC50 > 100000 nM T99989 C8VJY4 59406955 IC50 = 26 nM T99989 CPU7N9 60196195 IC50 = 260 nM T99989 CV63UL 67240318 IC50 > 10000 nM T99989 C29XOR 68517752 IC50 = 70 nM T99989 CP1L8B 68518789 IC50 = 1 nM T99989 C1WH7K 70679288 IC50 = 199 nM T99989 C2XV4Q 70694953 IC50 > 100000 nM T99989 CL1HY5 71212233 IC50 > 100000 nM T99989 CKX52R 71212291 IC50 > 100000 nM T99989 C0T2VB 71212317 IC50 = 50000 nM T99989 C5B8NS 71212337 IC50 > 100000 nM T99989 CSN04E 71212395 IC50 > 100000 nM T99989 C1OCW0 71212403 IC50 > 100000 nM T99989 CBX2I4 71212419 IC50 > 100000 nM T99989 CLS4R3 71212434 IC50 > 100000 nM T99989 CTF8M7 71212446 IC50 > 100000 nM T99989 C2Z8CX 71212514 IC50 > 100000 nM T99989 CBT7L3 71212517 IC50 > 100000 nM T99989 CHY91V 71578307 IC50 > 100000 nM T99989 C0W2KX 71578373 IC50 > 100000 nM T99989 C6TX9R 71578374 IC50 > 100000 nM T99989 C2D1RN 71578375 IC50 > 100000 nM T99989 C73MEW 71578445 IC50 = 20000 nM T99989 C5NH3V 71578446 IC50 = 80000 nM T99989 CC65WU 71578447 IC50 > 100000 nM T99989 CIP6Q2 71578520 IC50 > 100000 nM T99989 CPJ19D 71578658 IC50 > 100000 nM T99989 C5W0GC 71578744 IC50 > 100000 nM T99989 CLZ59B 71578745 IC50 > 100000 nM T99989 CHGS40 71710904 IC50 = 67.2 nM T99989 C67RXJ 71716255 IC50 = 4120 nM T99989 C8VE2W 72695133 IC50 = 190 nM T99989 C79APU 72720814 IC50 = 600 nM T99989 CK18UV 72720816 IC50 = 460 nM T99989 C9K7PA 72721921 IC50 = 160 nM T99989 C7V5NW 73265159 IC50 = 115 nM T99989 CIJ3M8 73293373 IC50 = 81.6 nM T99989 C91YZL 74396249 IC50 = 15.7 nM T99989 CJ35EI 78333498 IC50 = 500 nM T99989 CFA78Z 118117059 IC50 = 420 nM T99989 CU84JB 118117109 IC50 > 10000 nM T99989 CRP3J9 118117224 IC50 = 620 nM T99989 C9SF2U 118117741 IC50 = 320 nM T99989 CR5C6P 118135794 IC50 = 990 nM T99989 CFAE24 127042448 IC50 = 32.6 nM T99989 CA5XE4 129012139 IC50 <= 100 nM T99989 CH2S1Y 130431660 IC50 <= 100 nM T99989 C0BSA1 145963824 IC50 = 1145 nM T99989 CW05TY 145963985 IC50 = 1765 nM T99989 CBT15C 145964197 IC50 = 975 nM T99989 CD9FX7 145964328 IC50 = 1310 nM T99989 CPTW53 145964369 IC50 = 170 nM T99989 CN59FX 145964414 IC50 = 395 nM T99989 C4AR0G 145964627 IC50 = 1410 nM T99989 C3J6YH 145965218 IC50 = 280 nM T99989 CW12OV 145965254 IC50 = 54 nM T99989 CI39VD 145965319 IC50 = 370 nM T99989 C6ZW7D 145965387 IC50 = 250 nM T99989 C45SDT 145965497 IC50 = 385 nM T99989 CWK36T 145965775 IC50 = 1230 nM T99989 CB8VS5 145965873 IC50 = 2095 nM T99989 C0LM9U 145966033 IC50 = 375 nM T99989 C76NKD 145966367 IC50 = 50 nM T99989 CB8J9L 145966621 IC50 = 655 nM T99989 C5D7LE 145966696 IC50 = 320 nM T99989 CMJ31A 145966880 IC50 = 245 nM T99989 C4K2MZ 145967302 IC50 = 255 nM T99989 C8U7EA 145967475 IC50 = 1230 nM T99989 C6IZ1C 145967749 IC50 = 1905 nM T99989 C0ZML5 145967991 IC50 = 2955 nM T99989 C5I8UB 145968214 IC50 = 340 nM T99989 CO06FU 145968732 IC50 = 2010 nM T99989 C89WUQ 145969180 IC50 = 245 nM T99989 C93CMJ 145970268 IC50 = 125 nM T99989 CD6J3O 145970533 IC50 = 105 nM T99989 CZI5A9 145970735 IC50 = 630 nM T99989 C2O1ZW 145970740 IC50 = 385 nM T99989 COG2B8 145971011 IC50 = 315 nM T99989 CK03FQ 145972343 IC50 = 660 nM T99989 CAJ0D4 145972722 IC50 = 860 nM T99989 CWB10V 145973036 IC50 = 205 nM T99989 C3P1OT 145973084 IC50 = 135 nM T99989 CG48AP 145973222 IC50 = 16 nM T99989 CYC0U9 145973723 IC50 = 1840 nM T99989 CV2R6L 145973925 IC50 = 1195 nM T99989 C3UK4Q 145973964 IC50 = 335 nM T99989 CW0Y2I 145974384 IC50 = 205 nM T99989 C2YQN3 145974395 IC50 = 660 nM T99989 CH9LZ0 145974411 IC50 = 150 nM T99989 CKES90 145974470 IC50 = 990 nM T99989 CQR37C 145974951 IC50 = 265 nM T99989 C1N0DI 145975378 IC50 = 915 nM T99989 C1PSC3 145975405 IC50 > 10000 nM T99989 CPGZ90 145975408 IC50 = 105 nM T99989 CWF6C7 145976053 IC50 = 310 nM T99989 CSH68V 145976072 IC50 = 205 nM T99989 C43TWQ 145976109 IC50 = 715 nM T99989 C18QUZ 145976185 IC50 = 6560 nM T99989 CY2IN5 145976421 IC50 = 145 nM T99989 C9T0SR 145976580 IC50 = 560 nM T99989 CUP7F4 145976617 IC50 = 305 nM T99989 CLI3T5 145977030 IC50 = 380 nM T99989 CGV9W7 145977170 IC50 = 175 nM T99989 CJ2UR4 145977480 IC50 = 860 nM T99989 CA7S8J 145977657 IC50 > 10000 nM T99989 CU5L2G 145977991 IC50 > 10000 nM T99989 CMG04P 145978001 IC50 = 80 nM T99989 CS3ID1 145978144 IC50 = 1200 nM T99989 D00JGL 6419753 IC50 = 338 nM T99989 D04ZWF 53396311 IC50 > 5000 nM T99989 D06QYR 53472153 IC50 = 32 nM T99989 D0Q3KS 9957049 IC50 > 10000 nM T99989 D0UN8H 5288600 IC50 = 1000 nM T25663 CJM28K 453479 Ki = 42500 nM T25663 C7TF3A 51112335 EC50 = 8709.64 nM T25663 CPQL51 56783276 EC50 = 61659.5 nM T25663 C5NHJ0 72141742 EC50 = 5128.61 nM T25663 D00SDJ 11237664 IC50 > 10000 nM T25663 D01QYQ 6603931 EC50 = 67608.3 nM T40491 CN31KS 44372867 IC50 > 1000000 nM T40491 C71TJL 73351415 IC50 = 304 nM T40491 C32MLF 145964099 IC50 = 900 nM T40491 D01SLG 446512 IC50 = 7 nM T94094 D05RQB 457964 IC50 = 400 nM T94094 CZP5J2 3415 IC50 = 2500 nM T94094 CQ87XE 72187 IC50 = 22100 nM T94094 CU3P0Y 484047 IC50 = 400 nM T94094 C61SXL 492406 IC50 = 700 nM T94094 CZ1A8T 503580 IC50 = 1100 nM T94094 C69CXQ 6482388 IC50 = 2700 nM T94094 CTNS15 6482389 IC50 = 1000 nM T94094 CP3KF8 6482390 IC50 = 4200 nM T94094 CW0CT2 6482391 IC50 = 1100 nM T94094 C8J5HU 6482392 IC50 = 1800 nM T94094 CO27IL 6482393 IC50 = 2200 nM T94094 C8F1DN 6482394 IC50 = 400 nM T94094 CDQ5G3 6482395 IC50 = 670 nM T94094 CX97RA 6482396 IC50 = 2400 nM T94094 C65VNZ 6482397 IC50 = 750 nM T94094 CG42KR 6482398 IC50 = 810 nM T94094 CBX60C 6482399 IC50 = 18500 nM T94094 CZC8L3 6482400 IC50 = 4000 nM T94094 C91RUD 6482401 IC50 = 430 nM T94094 CZ32BN 6482402 IC50 = 9700 nM T94094 CEH67F 6482403 IC50 = 9500 nM T94094 CH8QA3 6482404 IC50 = 22000 nM T94094 C1U6KS 6483693 IC50 = 1800 nM T94094 CI5U3R 9870496 IC50 = 37 nM T94094 CS4FE9 9953786 IC50 = 1100 nM T94094 CW1KA2 9983320 IC50 = 200 nM T94094 CYPA38 10029378 IC50 = 100 nM T94094 CF5Q8X 10053197 IC50 = 65 nM T94094 CRA7U0 10368624 IC50 = 100 nM T94094 CE7N9R 10391097 IC50 = 100 nM T94094 C3OHC4 10391188 IC50 = 85 nM T94094 CK87ZA 10458488 IC50 = 100 nM T94094 CUR07A 11156325 IC50 = 175 nM T94094 CA2TU8 11202565 IC50 = 77 nM T94094 CS5V8Y 11237405 IC50 = 235 nM T94094 CQ89ME 11272615 IC50 = 12 nM T94094 C8UQ3G 11283149 IC50 = 250 nM T94094 CU0PL8 16729641 IC50 = 8400 nM T94094 C9G0AH 16729642 IC50 = 240 nM T94094 C6DNA5 16729643 IC50 = 1580 nM T94094 CVYL91 16729644 IC50 = 2040 nM T94094 CD97KH 16729645 IC50 = 8900 nM T94094 C5Q0DG 16729648 IC50 = 66 nM T94094 C9T5DU 16729649 IC50 = 315 nM T94094 C38VQU 16729650 IC50 = 87 nM T94094 CFJ1Y0 16729651 IC50 = 3530 nM T94094 CO0V9R 16729652 IC50 = 17500 nM T94094 C2U6QJ 16729653 IC50 = 2550 nM T94094 CUR2N6 44440867 IC50 = 220 nM T94094 C7IF5L 44440869 IC50 = 203 nM T94094 CJL29M 44440870 IC50 = 86 nM T94094 C3HGT2 44440871 IC50 = 160 nM T94094 CL9B0C 44440875 IC50 = 35 nM T94094 C6IZ1X 44440876 IC50 = 200 nM T94094 CJW15U 44440877 IC50 = 180 nM T94094 C4YZO1 44440878 IC50 = 350 nM T94094 C17GVK 44440879 IC50 = 240 nM T94094 CFE5M1 44440880 IC50 = 280 nM T94094 CO6EH7 44440881 IC50 = 61 nM T11072 D00XWD 135409453 Ki < 100 nM T11072 D01AZG 5073 Ki = 1000 nM T11072 D01TSI 8223 Ki = 0.8 nM T11072 D03RZV 5504 Ki > 10000 nM T11072 D06FPQ 77992 Ki = 4.4 nM T11072 D08VRO 3822 IC50 = 260 nM T11072 D09EBS 4636 Ki = 0.4 nM T11072 D0CQ0Z 33630 Ki = 3560 nM T11072 D0G8NN 119570 Ki > 10000 nM T11072 D0H3HM 60795 Ki = 100 nM T11072 D0H7KF 5002 Ki > 1000 nM T11072 D0NG7O 60857 Ki = 0.76 nM T11072 D0R6RO 4184 IC50 = 380.19 nM T11072 D0S9MU 5078 EC50 = 3 nM T11072 D0T3KI 4440 EC50 = 1.6 nM T11072 D0V4QS 135398745 Ki > 1000 nM T11072 D0WV3U 4893 Ki = 0.33 nM T11072 D0Y4DY 5709 Ki = 0.7 nM T11072 D0Z1RV 135398737 Ki > 1000 nM T11072 D0Z6UC 5358 Ki = 1.2 nM T11072 D04GMY 11842633 Ki < 100 nM T11072 D08CJK 1150 Ki = 23 nM T11072 D09GHO 5311258 Ki = 137 nM T11072 D0N1HW 5311200 Ki > 10000 nM T11072 D0X2XF 177336 Ki < 10000 nM T11072 D00OWF 5280953 Ki > 10000 nM T11072 D00NLD 9881526 IC50 = 0.3 nM T11072 D02ZSO 6426760 IC50 = 0.6 nM T11072 D03PJW 108029 IC50 = 39 nM T11072 D03SWH 9845148 Ki = 4.6 nM T11072 D06DZI 107780 Ki = 0.1259 nM T11072 D08AWI 11430856 Ki > 2000 nM T11072 D08XWZ 9860595 Ki = 8 nM T11072 D0B7SP 11292933 Ki = 0.1995 nM T11072 D0M7LV 5761 Ki = 3.9 nM T11072 D0SU1F 132552 IC50 = 7.244 nM T11072 D0T1SF 9909448 Ki = 0.9 nM T11072 D0U7VZ 11225102 Ki < 100 nM T11072 D0Y0RW 66004 IC50 = 2.512 nM T11072 D0YP7L 6604889 Ki = 1584.89 nM T11072 C5JG6U 2689 IC50 = 35 nM T11072 C32BCH 4656 Ki = 50 nM T11072 C5H9CN 9287 Ki = 1790 nM T11072 C6Y7RT 15760 Ki = 6.4 nM T11072 CVD75F 20810 Ki = 9.7 nM T11072 CW3PK7 26395 IC50 = 77 nM T11072 C0OZ3N 37732 Ki = 1800 nM T11072 C6WDL7 49756 Ki = 250 nM T11072 CTB26S 52899 Ki = 1060 nM T11072 C8UPV1 59022 IC50 = 25 nM T11072 CAF7T8 64622 Ki = 460 nM T11072 CW2T4Y 78576 Ki = 2075 nM T11072 CN9GK1 104911 Ki > 10000 nM T11072 CKP25M 121881 Ki < 10000 nM T11072 CFSE35 129503 Ki = 12 nM T11072 C4PR2E 132564 IC50 = 4200 nM T11072 CD89VU 137235 Ki > 30000 nM T11072 CGT8R0 160510 Ki > 10000 nM T11072 CF3US2 169764 IC50 = 820 nM T11072 CZ3N4E 178081 Ki = 173 nM T11072 COPZ85 188006 Ki = 3.7 nM T11072 CQ97BV 225047 Ki > 10000 nM T11072 CYV1R3 417052 Ki > 10000 nM T11072 C2VLP8 752521 Ki = 2655 nM T11072 C7Y3LQ 1328538 Ki = 590 nM T11072 C5DU2K 2199302 Ki = 34 nM T11072 C7PM8O 2261792 Ki = 68 nM T11072 CNMB94 2574642 Ki = 1360 nM T11072 CMP82C 2762736 Ki = 0.6 nM T11072 CB3M6V 2762737 Ki = 0.4 nM T11072 C3M7GN 3016908 Ki = 72 nM T11072 CAM8H3 3066250 IC50 > 1000 nM T11072 CS8KE2 3649661 Ki = 8590 nM T11072 C2A4KH 4202024 Ki = 3.4 nM T11072 CW34VC 6160690 Ki = 0.3 nM T11072 C9EO4Z 6422277 Ki = 112 nM T11072 CZV19U 6426761 EC50 = 0.7 nM T11072 CXZ53N 6603866 Ki = 164 nM T11072 C3A1FO 6604789 Ki = 39810.72 nM T11072 C0QCK1 6918455 Ki = 251.19 nM T11072 CW0ZE5 6918542 Ki = 720 nM T11072 CC5PQ0 6918601 Ki = 3900 nM T11072 C1WXY3 6918603 Ki = 630.96 nM T11072 CD0Z4I 6918648 Ki = 199.53 nM T11072 C8AL9V 6918689 Ki < 100000 nM T11072 CCT52F 9795333 Ki = 74 nM T11072 C71EYQ 9796492 EC50 = 0.3 nM T11072 CUD06Z 9796627 Ki = 180 nM T11072 CX7I8J 9802187 Ki = 8 nM T11072 C2MOX8 9802224 Ki = 27 nM T11072 CCV0M4 9802530 Ki = 3.2 nM T11072 CZL0O6 9803620 IC50 = 5.4 nM T11072 CE0DI5 9804612 Ki = 79.43 nM T11072 CNX4F0 9805456 Ki = 398.11 nM T11072 CPZ05H 9805881 Ki = 1.3 nM T11072 CGJB47 9816035 Ki = 6.8 nM T11072 CH7U3C 9816604 Ki = 86 nM T11072 C0WKI4 9817415 Ki = 3.4 nM T11072 CWOS30 9817810 Ki = 4.5 nM T11072 CX7N8J 9817881 IC50 = 3.162 nM T11072 CWS18C 9832057 Ki = 0.89 nM T11072 C3K4XT 9837108 Ki = 340 nM T11072 CRW5N0 9837525 Ki = 1.1 nM T11072 C53UPQ 9842861 Ki = 5000 nM T11072 C28HXY 9844873 EC50 = 0.4 nM T11072 CC24WR 9845261 IC50 = 700 nM T11072 CS1ID2 9846928 IC50 = 3 nM T11072 CYMP40 9851789 IC50 = 0.05 nM T11072 CM13ZV 9856041 Ki = 1900 nM T11072 CNCK78 9862256 Ki = 9.3 nM T11072 C8M5XK 9863333 Ki = 6.7 nM T11072 C8ROC3 9866484 EC50 = 7.5 nM T11072 CB1F0C 9867475 Ki = 98 nM T11072 C57YPX 9867902 EC50 = 3.5 nM T11072 C7AB8O 9870053 Ki = 2511.89 nM T11072 C19VUG 9871977 Ki = 398.11 nM T11072 C1WF3D 9881478 Ki = 1190 nM T11072 CZ6NK9 9881603 Ki = 33 nM T11072 COW86S 9886269 Ki = 2650 nM T11072 CJW1P5 9888494 Ki = 2398.83 nM T11072 C6N8UE 9889681 Ki = 158.49 nM T11072 CM52WU 9890119 Ki = 199.53 nM T11072 CF5GN4 9890331 IC50 = 2.5 nM T11072 CEG1K5 9891002 Ki = 398.11 nM T11072 C7QMK5 9891617 Ki = 316.23 nM T11072 CEL29O 9891618 Ki = 251.19 nM T11072 C3J8GU 9892409 Ki = 316.23 nM T11072 CFM67S 9897637 Ki = 0.45 nM T11072 CFI97S 9904205 IC50 = 660.69 nM T11072 CUN81Q 9905249 Ki > 10000 nM T11072 CYWQ50 9906447 Ki = 6380 nM T11072 CYZ5N4 9909089 Ki = 0.1585 nM T11072 C78MDV 9913554 Ki = 100 nM T11072 C4UYZ7 9927441 Ki = 510 nM T11072 CJ6CF2 9928474 Ki = 16 nM T11072 CJS2T1 9930155 IC50 = 6.3 nM T11072 CYVZ47 9934284 Ki = 251.19 nM T11072 CWO45F 9935387 Ki = 125.89 nM T11072 CYH3R7 9947817 Ki = 730 nM T11072 C41HSL 9948210 Ki = 155 nM T11072 CM5A2D 9949172 IC50 = 33 nM T11072 CN7A4C 9949568 Ki = 30 nM T11072 C63EWV 9950390 Ki = 3100 nM T11072 CP5MQ0 9950538 IC50 = 1.3 nM T11072 CO49NV 9952249 EC50 = 0.6 nM T11072 CK8NR2 9954121 Ki = 1258.93 nM T11072 C48OKD 9954663 Ki = 21 nM T11072 C9QPM4 9955522 Ki = 0.631 nM T11072 CSK1B2 9955819 Ki = 0.69 nM T11072 CFR41N 9957068 Ki = 1258.93 nM T11072 CZ9SC7 9957274 Ki = 0.631 nM T11072 CGO64P 9957376 Ki = 0.1995 nM T11072 CTZ4U0 9972838 Ki = 108 nM T11072 CYK05G 9973090 Ki = 18 nM T11072 C2XG1I 9977716 Ki = 0.1995 nM T11072 CFN50J 9978683 Ki > 5000 nM T11072 CPX92V 9979309 Ki = 0.1 nM T11072 CXZM08 9981270 Ki = 9.8 nM T11072 CDG74Q 9983460 Ki = 0.26 nM T11072 CCR0T4 9984109 Ki = 0.42 nM T11072 CN3D8M 9994674 Ki = 7.5 nM T11072 C1RNF9 9995233 Ki = 7.6 nM T11072 CXI19F 9997421 Ki = 87 nM T11072 CSGQ91 9997422 Ki = 54 nM T11072 CWQ1K3 9999722 Ki = 0.4 nM T11072 C8A6EZ 10001971 Ki = 0.3981 nM T11072 CVWG72 10003116 Ki = 1.4 nM T11072 CCE86A 10003971 Ki = 5 nM T11072 CV4T9U 10008868 Ki = 0.09 nM T11072 C3S7XA 10009042 IC50 = 0.11 nM T11072 C4F5JB 10015980 Ki = 16 nM T11072 CV7IP3 10016747 Ki = 3.2 nM T11072 C8JFH0 10016864 Ki = 26 nM T11072 CV7R9F 10020040 Ki > 10000 nM T11072 CK18LT 10020895 Ki = 730 nM T11072 C04ZAS 10021450 Ki = 2.8 nM T11072 CQHW51 10023176 Ki = 0.2512 nM T11072 CM7W9G 10024936 Ki = 10 nM T11072 C2EUY0 10035109 Ki > 10000 nM T11072 CA7MG0 10044965 Ki = 2 nM T11072 C4S0HI 10047915 Ki = 0.3 nM T11072 C2JZL1 10048222 Ki = 0.52 nM T11072 C2UI7F 10048252 Ki = 3.6 nM T11072 CF84QJ 10048342 Ki = 0.3981 nM T11072 C8JLO2 10048343 Ki = 12.59 nM T11072 C5PQ2I 10060289 Ki = 1.6 nM T11072 C9ENY6 10062659 Ki = 14 nM T11072 CHQ1L3 10064361 Ki = 34 nM T11072 C0GI7T 10064500 Ki = 192 nM T11072 C98DKQ 10065239 Ki = 419 nM T11072 C6DC9G 10065919 Ki = 440 nM T11072 C2EG0W 10068933 Ki = 540 nM T11072 CXW80P 10069802 Ki = 3.4 nM T11072 C6HP2C 10069977 Ki = 1.8 nM T11072 CJM76I 10070281 Ki = 5.4 nM T11072 C9KWT3 10071738 Ki = 0.1585 nM T11072 CV6R2F 10073139 Ki = 12.59 nM T11072 CQ1YA4 10076876 Ki = 3.9 nM T11072 CIO9D1 10088038 Ki = 8.4 nM T11072 C2M6UR 10088426 Ki = 125 nM T11072 C9OXA7 10095692 Ki = 1250 nM T11072 CIZ50V 10096890 Ki = 0.88 nM T11072 C54EYD 10108561 IC50 < 1000 nM T11072 C2ISY6 10114480 Ki = 2.512 nM T11072 C9PG3D 10115847 Ki = 63.1 nM T11072 CJZX05 10115848 Ki = 794.33 nM T11072 CP1CL5 10127149 Ki = 6.31 nM T11072 CLFA47 10127209 Ki = 2511.89 nM T11072 CKYQ52 10127424 Ki = 1 nM T11072 CRJ8M9 10127673 Ki = 1 nM T11072 C4SN0A 10127877 Ki = 0.631 nM T11072 C9J6KH 10128059 Ki = 6.31 nM T11072 CNA8W3 10130620 Ki = 105 nM T11072 CXCY91 10131024 Ki = 0.97 nM T11072 CWMT35 10138727 Ki = 398.11 nM T11072 C4X9RB 10150658 Ki = 1.585 nM T11072 CKGC73 10150796 Ki = 0.2512 nM T11072 CJI9T7 10151492 Ki = 0.2512 nM T11072 CSPG27 10159927 Ki = 10 nM T11072 C9JLX2 10161027 Ki = 79.43 nM T11072 CVA6N0 10161028 Ki = 3.162 nM T11072 C5E4SQ 10172853 Ki = 2.512 nM T11072 C3YT8A 10173169 Ki = 2.512 nM T11072 CJRV76 10173263 Ki = 0.5012 nM T11072 CMP89S 10173443 Ki = 2.512 nM T11072 CT0CX5 10174078 Ki = 0.7943 nM T11072 CQXI36 10174088 Ki = 1.585 nM T11072 C34ROH 10174199 Ki = 0.3981 nM T11072 CEDP29 10183895 Ki = 3.981 nM T11072 C6NA5G 10194297 Ki = 3.162 nM T11072 CI76JU 10194809 Ki = 0.631 nM T11072 CLHY30 10194820 Ki = 0.3162 nM T11072 CW1CM3 10195275 Ki = 0.5012 nM T11072 CNT0Y6 10198320 Ki = 13 nM T11072 CMWD23 10198756 Ki = 23 nM T11072 CE3S6M 10216160 Ki = 3.162 nM T11072 CRW49L 10216744 Ki = 7.943 nM T11072 C80QXD 10216873 Ki = 1.995 nM T11072 CQ7ND4 10220230 Ki = 420 nM T11072 CF4N1M 10237964 Ki = 0.5012 nM T11072 C0Q2ZD 10238160 Ki = 3.981 nM T11072 CIR98N 10238565 Ki = 1 nM T11072 CK39BA 10238566 Ki = 0.631 nM T11072 C3L0WD 10238762 Ki = 3.981 nM T11072 CI9KH6 10238763 Ki = 10 nM T11072 CK5TC1 10243466 Ki = 170 nM T11072 C6K5ZM 10244251 IC50 = 9300 nM T11072 CC36JL 10245352 Ki = 63 nM T11072 CVF1E5 10246054 IC50 > 1000 nM T11072 CK9NT0 10247448 Ki = 54 nM T11072 C4Q2SH 10249573 Ki = 630.96 nM T11072 CMA42P 10250834 Ki = 0.93 nM T11072 CD83JK 10251722 Ki = 48 nM T11072 CUSP67 10252256 EC50 = 1.7 nM T11072 C2JDW3 10253939 Ki = 1.8 nM T11072 CX67OE 10254537 Ki = 0.34 nM T11072 CRNC25 10265814 Ki = 75 nM T11072 C7DJ2O 10266598 Ki = 19 nM T11072 CH31DX 10267394 Ki > 10000 nM T11072 CTE91S 10267412 Ki = 24 nM T11072 CVC87R 10275633 Ki = 0.3981 nM T11072 CQ8N3F 10288132 Ki = 1 nM T11072 C3G8KJ 10310285 Ki = 1.995 nM T11072 C0WRV9 10310423 Ki = 2.512 nM T11072 CU89JD 10314060 Ki > 10000 nM T11072 C0OJ2C 10319235 Ki = 0.1585 nM T11072 C7BI8J 10319498 EC50 = 0.5 nM T11072 CPH30X 10319737 Ki = 0.3162 nM T11072 CCXJ27 10321497 Ki = 0.31 nM T11072 CISG65 10323598 IC50 = 37 nM T11072 C30CBI 10324625 Ki = 1.3 nM T11072 CP52QF 10331989 Ki = 19 nM T11072 C3E5CB 10337773 Ki < 100000 nM T11072 CM10QP 10340549 Ki = 1.64 nM T11072 CXG6B1 10341129 Ki = 0.3162 nM T11072 C4IA8Z 10341917 EC50 = 0.9 nM T11072 C0UTS5 10342552 Ki = 0.31 nM T11072 C3ZN0F 10344705 Ki = 0.56 nM T11072 C9IAV3 10346043 Ki > 1584.89 nM T11072 CS24DU 10353268 IC50 = 110 nM T11072 CWON13 10354282 Ki = 77 nM T11072 CG0X4W 10356544 Ki = 43 nM T11072 CL9H5K 10358173 Ki = 6.5 nM T11072 C2J3OP 10358224 Ki = 8.6 nM T11072 CR03MZ 10360150 Ki = 36 nM T11072 CR53YS 10365683 Ki = 1.4 nM T11072 CM97GO 10370874 Ki = 100 nM T11072 C1P9DA 10376496 Ki = 69 nM T11072 CW7MQ0 10376578 EC50 = 0.22 nM T11072 C5T7AE 10378357 Ki = 35 nM T11072 CPU8B2 10379784 Ki = 42 nM T11072 CDAC63 10381889 IC50 = 134.9 nM T11072 CM47BF 10382523 Ki = 13 nM T11072 C36TNW 10383010 Ki = 33 nM T11072 CMZA83 10383646 Ki > 5000 nM T11072 C69KIB 10385855 EC50 = 0.6 nM T11072 C0XG9M 10387420 Ki = 0.2512 nM T11072 C1U7LS 10398118 Ki = 585 nM T11072 C20KTU 10400189 Ki = 27 nM T11072 C3ESO4 10401862 Ki = 294 nM T11072 CQ5V6K 10402263 Ki = 6.7 nM T11072 CG60RT 10403260 Ki = 334 nM T11072 C9RZ1N 10403999 Ki = 2.5 nM T11072 CLEU45 10406614 Ki = 2 nM T11072 CMBW49 10408880 Ki = 0.39 nM T11072 C4TPN1 10413595 Ki = 199.53 nM T11072 C2B0IU 10421236 Ki > 10000 nM T11072 CK1WH6 10424220 Ki = 11 nM T11072 CQ2Y4A 10425027 Ki = 217 nM T11072 CR4LS0 10430623 Ki > 5000 nM T11072 CN58XF 10432512 Ki = 5.1 nM T11072 CD7U5I 10433930 Ki > 3162.28 nM T11072 CDU91R 10434550 Ki = 26 nM T11072 CBAY90 10445946 Ki = 250 nM T11072 CCY68S 10448470 Ki = 4.4 nM T11072 C9S5WP 10449461 Ki = 7.4 nM T11072 C9WA5Q 10452875 Ki = 0.2512 nM T11072 CFK16Y 10454806 Ki = 0.3981 nM T11072 CYMS64 10454807 Ki = 0.1995 nM T11072 C62WSQ 10456474 Ki = 1.2 nM T11072 C57RFG 10456869 IC50 = 1.2 nM T11072 C8V6ZQ 10458087 Ki = 1 nM T11072 CQ4T7G 10458088 Ki = 0.53 nM T11072 CYS76Z 10468376 Ki = 440 nM T11072 COV85C 10472143 Ki = 2.4 nM T11072 C73TEG 10475893 Ki = 13 nM T11072 CCRX82 10476740 EC50 = 1.2 nM T11072 CL63TF 10477223 Ki = 0.1995 nM T11072 C8JCZ1 10477386 Ki = 0.42 nM T11072 CE9R8Z 10477461 IC50 = 0.65 nM T11072 CWY2J3 10478217 Ki = 0.1995 nM T11072 CEF2O6 10478367 Ki = 105.9 nM T11072 CPB1I5 10488933 Ki = 2520 nM T11072 C1XT2J 10490160 Ki = 4390 nM T11072 CI7D5J 10490521 Ki = 0.44 nM T11072 CVJ4I3 10494885 IC50 = 64.57 nM T11072 C0I3BG 10496545 Ki = 2350 nM T11072 CQ9A2N 10498633 Ki = 223 nM T11072 C65KTM 10500370 IC50 = 9.1 nM T11072 C4IXZ5 10500422 Ki = 169 nM T11072 C9SV3J 10501944 EC50 = 1.5 nM T11072 C97AGV 10501945 IC50 = 0.72 nM T11072 C74XEH 10502669 EC50 = 0.3 nM T11072 CNGM74 10502763 EC50 = 1.8 nM T11072 C1ALS8 10502988 EC50 = 4.2 nM T11072 CD3IL2 10503687 IC50 = 0.7 nM T11072 CD47NC 10503731 EC50 = 0.6 nM T11072 CCM78N 10504095 EC50 = 15 nM T11072 CS1RN9 10504096 IC50 = 4.3 nM T11072 CY7OA9 10504097 EC50 = 3.4 nM T11072 CNUR81 10504600 IC50 = 1.5 nM T11072 C2FDP8 10505438 IC50 = 6.9 nM T11072 CFJ45P 10505525 IC50 = 1.5 nM T11072 CUT89L 10517352 Ki = 1098 nM T11072 CCPO93 10518850 Ki = 2.8 nM T11072 CNAZ85 10519108 IC50 = 26 nM T11072 CCQA42 10525100 IC50 = 3.8 nM T11072 CT28NZ 10526567 EC50 = 12 nM T11072 CP16JO 10526642 IC50 = 8.3 nM T11072 CUWV98 10526736 IC50 = 0.5 nM T11072 CF47AX 10526737 IC50 = 6.8 nM T11072 CSNQ16 10527410 Ki = 1318.26 nM T11072 CA15PT 10527882 EC50 = 1 nM T11072 CZLC18 10528410 IC50 = 5.9 nM T11072 CYP31J 10530932 IC50 > 1000 nM T11072 C0ZM5P 10531639 Ki = 0.27 nM T11072 C5HEN4 10536129 Ki = 2375 nM T11072 CI36TG 10539089 IC50 = 14.79 nM T11072 CE3OX5 10541847 Ki = 1095 nM T11072 CF8NY5 10546537 IC50 = 338.84 nM T11072 CN3EP8 10548444 IC50 = 1.6 nM T11072 CIKZ61 10549785 IC50 = 35 nM T11072 C8AC6N 10550488 EC50 = 18 nM T11072 CNR5F7 10550857 IC50 = 0.1 nM T11072 CYB74T 10551206 IC50 = 1.4 nM T11072 CXA12U 10551207 IC50 = 5.5 nM T11072 C4MP8V 10551328 IC50 = 0.6 nM T11072 C3UK0W 10551525 IC50 = 4.7 nM T11072 C8CGV9 10551857 IC50 = 4.5 nM T11072 CL9O3W 10552243 EC50 = 4.7 nM T11072 CUE54L 10552573 EC50 = 6 nM T11072 CX0N3A 10552663 IC50 = 1.5 nM T11072 CHOZ29 10567450 Ki = 42 nM T11072 CP53ZW 10571716 IC50 = 20 nM T11072 CJ2YD5 10572483 IC50 = 1.5 nM T11072 CP7AX5 10573843 IC50 = 1 nM T11072 CHE80N 10573876 Ki = 501.19 nM T11072 C4Y1WU 10573904 IC50 = 1.7 nM T11072 CVI9U2 10574570 EC50 = 0.3 nM T11072 CMX1B0 10574671 IC50 = 0.8 nM T11072 CIB5V0 10574762 IC50 = 0.8 nM T11072 C5CR0T 10575553 IC50 = 3.5 nM T11072 CJC3R5 10575878 IC50 = 12 nM T11072 CWPE61 10576874 IC50 = 19 nM T11072 C09ZXH 10577268 Ki = 25.12 nM T11072 CA8NT1 10577311 EC50 = 2.8 nM T11072 CG85VM 10578117 IC50 = 600 nM T11072 CWM6U4 10588458 Ki = 143 nM T11072 C1O3LZ 10588665 IC50 = 14.45 nM T11072 CCBU34 10590370 Ki = 210 nM T11072 C0N2EP 10592083 IC50 = 12 nM T11072 CY3BD0 10592324 IC50 = 28.84 nM T11072 CJV2Z4 10596387 EC50 = 31 nM T11072 CITF30 10596566 EC50 = 0.3 nM T11072 CO23YX 10597140 Ki = 501.19 nM T11072 C6I3LK 10597210 Ki = 39.81 nM T11072 C4Y2OD 10597901 IC50 = 4.8 nM T11072 CE3W5U 10597902 EC50 = 3 nM T11072 CW25KM 10600063 EC50 = 3.2 nM T11072 CKJZ76 10600212 IC50 = 1 nM T11072 C98XYU 10600213 IC50 = 1 nM T11072 CJ3F2B 10600678 IC50 = 1.4 nM T11072 C5X7BD 10600871 IC50 = 467 nM T11072 CKH1P3 10601144 IC50 = 5 nM T11072 CF74VT 10601619 Ki = 0.62 nM T11072 CC9B5J 10602052 IC50 = 8.1 nM T11072 C0LRY1 10612178 IC50 = 724.44 nM T11072 CVYB63 10613373 Ki = 1.6 nM T11072 C1UVB3 10614906 EC50 = 80 nM T11072 CCVT79 10614907 IC50 = 31 nM T11072 CF5PK0 10617665 IC50 = 141.25 nM T11072 C8GFT6 10618751 Ki = 12 nM T11072 C06DSC 10620429 EC50 = 0.5 nM T11072 CX3A0P 10620719 Ki = 3.8 nM T11072 CWQ83M 10621020 IC50 = 37 nM T11072 CPF68U 10621021 EC50 = 0.1 nM T11072 CD8KX9 10621491 Ki = 298 nM T11072 CX09MP 10623434 IC50 = 5.5 nM T11072 CQO50M 10623614 EC50 = 1.3 nM T11072 C04NHF 10624003 IC50 = 35 nM T11072 C6K7IB 10624680 IC50 = 400 nM T11072 C8SN9G 10624768 Ki = 39.81 nM T11072 CN3H7E 10625408 IC50 = 18 nM T11072 C5R0MA 10627612 IC50 > 1000 nM T11072 CRB8C0 10635169 Ki = 82 nM T11072 C1MYD5 10640199 Ki = 69 nM T11072 C2FH3S 10643939 Ki = 560 nM T11072 C7R0EY 10643940 IC50 = 194.98 nM T11072 CLIA32 10644749 IC50 = 3.6 nM T11072 CQ98VE 10644750 EC50 = 0.3 nM T11072 CTM21V 10645471 EC50 = 0.9 nM T11072 C85DEQ 10645715 EC50 = 8.9 nM T11072 CDJ83U 10646873 IC50 = 4.4 nM T11072 CY7CU2 10646958 IC50 = 1.3 nM T11072 CPW89L 10646959 IC50 = 4.1 nM T11072 C0K2XA 10647181 IC50 = 1 nM T11072 C6PBY1 10647387 Ki = 0.35 nM T11072 CYDV92 10649124 Ki = 0.45 nM T11072 C4NW8J 10655811 Ki = 1900 nM T11072 CA3E2W 10664878 IC50 = 501.19 nM T11072 CNH98X 10665840 IC50 = 3090.3 nM T11072 CZ01DX 10667886 IC50 = 1.4 nM T11072 CTO51R 10670211 EC50 = 4 nM T11072 CB6YO4 10670534 IC50 = 0.4 nM T11072 C6XT1C 10670879 EC50 = 4.5 nM T11072 CR37GO 10671315 EC50 = 34 nM T11072 CVA06U 10671996 IC50 = 43 nM T11072 C0U6ZS 10672840 Ki = 0.88 nM T11072 C4BS9A 10673329 Ki = 5.012 nM T11072 C75AQY 10673854 IC50 = 700 nM T11072 C9U4LX 10679184 Ki > 10000 nM T11072 C8F1SI 10689227 IC50 = 17 nM T11072 C5FQ9T 10691904 Ki = 36 nM T11072 C9OHV5 10691928 IC50 = 22 nM T11072 C2LU1H 10692095 Ki = 238 nM T11072 COV35P 10693140 IC50 = 0.45 nM T11072 C2AI0W 10693206 IC50 = 2.1 nM T11072 CA3XK7 10693207 IC50 = 14 nM T11072 C4RN7E 10694177 IC50 = 78 nM T11072 C6AR7P 10694686 IC50 = 13 nM T11072 CSY6R8 10694810 IC50 = 56 nM T11072 CSJ83Y 10694895 IC50 = 280 nM T11072 CEIQ24 10695596 EC50 = 35 nM T11072 CYI47N 10696275 IC50 = 12 nM T11072 CM31PB 10696930 Ki = 0.3 nM T11072 COYX78 10709057 IC50 = 562.34 nM T11072 CE7DB9 10710400 Ki = 55 nM T11072 C97LJV 10714071 IC50 = 1479.11 nM T11072 CHW9D0 10716915 IC50 = 0.1 nM T11072 C3Y9FE 10717709 EC50 = 3.5 nM T11072 C4N7MI 10718668 EC50 = 10 nM T11072 C5G9PK 10718709 IC50 = 10 nM T11072 CG6A0Q 10718714 EC50 = 3.6 nM T11072 C15RUN 10719202 EC50 = 0.8 nM T11072 CYHQ97 10719203 IC50 = 3 nM T11072 CL1UQ7 10719245 IC50 = 6 nM T11072 CM9H8J 10719448 IC50 = 6.2 nM T11072 C3F7XV 10719687 EC50 = 0.2 nM T11072 CX8U7Y 10719938 IC50 = 1.6 nM T11072 C2Y5UQ 10720175 IC50 = 0.6 nM T11072 CUS3R0 10720301 Ki = 0.16 nM T11072 CTC31X 10733010 Ki = 10.8 nM T11072 C1FEW3 10733696 IC50 = 24 nM T11072 CAT6N3 10733823 IC50 = 8.8 nM T11072 C4M0JH 10738913 Ki = 10000 nM T11072 CH1PV5 10739818 EC50 = 2.1 nM T11072 C3PBD8 10740531 IC50 = 2.6 nM T11072 C2IK5A 10741528 IC50 = 0.5 nM T11072 CIA9Z0 10741826 EC50 = 2.2 nM T11072 C83YNJ 10753714 Ki = 6.2 nM T11072 C61VBM 10757342 IC50 = 933.25 nM T11072 CO0QF6 10759465 IC50 = 210 nM T11072 CLBQ57 10764284 IC50 = 173 nM T11072 CC49QS 10764869 IC50 = 0.7 nM T11072 CWYI16 10764998 IC50 = 0.35 nM T11072 CFXR10 10765655 EC50 = 0.9 nM T11072 C1I9OU 10766235 EC50 = 13 nM T11072 CNJ40K 10766277 IC50 = 18 nM T11072 CR2I0K 10766318 EC50 = 0.9 nM T11072 C2R0QI 10766319 EC50 = 5.1 nM T11072 CD7JC0 10766320 IC50 = 3.4 nM T11072 CJD70A 10766321 IC50 = 5.9 nM T11072 C8X2BM 10766570 EC50 = 1.9 nM T11072 C48HGI 10767140 IC50 = 1.8 nM T11072 CLDH19 10767244 IC50 = 4.2 nM T11072 CL5G7U 10768115 IC50 = 17 nM T11072 C54KOF 10768329 IC50 = 15 nM T11072 CP56UK 10774567 Ki = 1035 nM T11072 C9JW7S 10780344 EC50 = 7.8 nM T11072 CCB14F 10782381 IC50 = 2454.71 nM T11072 CZJO64 10782681 Ki = 42 nM T11072 CX70KH 10786335 Ki = 1200 nM T11072 CB6Q0L 10786628 IC50 = 9.8 nM T11072 CP3V4H 10787240 IC50 = 0.81 nM T11072 CW5L3X 10787241 EC50 = 9.5 nM T11072 C7RC5Y 10788620 IC50 = 4.2 nM T11072 CK34DX 10788768 EC50 = 0.3 nM T11072 C78QWE 10789334 IC50 = 1.1 nM T11072 CC48LD 10789399 IC50 = 0.9 nM T11072 CSDI98 10789717 IC50 = 5.8 nM T11072 CKG19X 10790076 EC50 = 14 nM T11072 C8Y3TP 10791125 Ki = 1.9 nM T11072 CNUF06 10791244 Ki = 0.35 nM T11072 C7GF8M 10791443 Ki = 19.95 nM T11072 CC6B1S 10799383 Ki = 1.7 nM T11072 CK9O3B 10802304 Ki = 4.9 nM T11072 C4VA1L 10805623 IC50 = 190 nM T11072 C4UR8Q 10805740 IC50 = 190.55 nM T11072 CXY1Q0 10809674 Ki = 1 nM T11072 CU2QG3 10811007 IC50 = 1.6 nM T11072 CH94VG 10811801 EC50 = 7.8 nM T11072 CW1Y5T 10811964 IC50 = 9.3 nM T11072 CIL3O6 10812465 IC50 = 1.6 nM T11072 CZG3J2 10812592 IC50 = 2 nM T11072 CRN89V 10812693 IC50 = 30 nM T11072 C8J2GW 10813272 EC50 = 0.5 nM T11072 CZT8S0 10813413 IC50 = 0.8 nM T11072 CA70HZ 10813769 EC50 = 30 nM T11072 C8NM9E 10814273 EC50 = 1.6 nM T11072 CW2LK3 10828231 Ki = 42 nM T11072 C78FDC 10834908 IC50 = 95 nM T11072 CY15OU 10834909 EC50 = 0.3 nM T11072 C8MHZ9 10835110 Ki = 630.96 nM T11072 CLE1W7 10835665 EC50 = 13 nM T11072 CMD47Q 10835928 IC50 = 2.6 nM T11072 CL2S9M 10836290 IC50 = 5.2 nM T11072 CF3W8J 10836301 IC50 = 4.2 nM T11072 C0MNA5 10836606 Ki = 0.46 nM T11072 C5L4HY 10836850 IC50 = 8.9 nM T11072 C30FNB 10836986 EC50 = 0.8 nM T11072 C2UJQ9 10837591 EC50 = 32 nM T11072 CHCV53 10837853 EC50 = 16 nM T11072 C83QOA 10837858 Ki = 0.4 nM T11072 CC8XL5 10838063 Ki = 0.51 nM T11072 C1ARP7 10838153 IC50 = 1.3 nM T11072 C1TI9X 10838622 IC50 = 29 nM T11072 C3IHO1 10838684 EC50 = 9.3 nM T11072 CCH9T7 10838923 Ki = 1995.26 nM T11072 C1OL4F 10839082 IC50 = 5.7 nM T11072 C98RSP 10847427 Ki > 10000 nM T11072 C4V3RT 10848041 Ki = 1.5 nM T11072 C6D1CX 10852406 IC50 = 2041.74 nM T11072 CIG0Y6 10858566 Ki = 16 nM T11072 CPLT37 10870264 Ki = 31 nM T11072 C8HN1F 10872581 Ki = 340 nM T11072 C8OYI0 10891048 Ki = 470 nM T11072 C1RAP3 10904295 Ki = 53 nM T11072 C6D7JR 10924369 Ki = 1470 nM T11072 CZN8J0 10925382 Ki = 930 nM T11072 C5X1OQ 10926112 Ki = 490 nM T11072 CWE3C9 10946905 Ki = 900 nM T11072 CNB39C 10947658 Ki = 3.7 nM T11072 C7GHU5 10970604 Ki = 3.8 nM T11072 C86GIP 10971452 Ki = 83 nM T11072 C51NOQ 10982183 Ki = 1122.02 nM T11072 C7O5UG 11003379 Ki = 170 nM T11072 CJS79L 11011968 Ki = 1800 nM T11072 CS0Z2D 11024311 Ki < 10000 nM T11072 CSU4T7 11024618 Ki = 1900 nM T11072 C4Y9XK 11033734 Ki = 80 nM T11072 CX73TF 11035452 Ki = 440 nM T11072 C7ID8S 11043914 Ki = 39 nM T11072 C3G0FH 11046087 Ki = 810 nM T11072 CG0J7X 11047115 Ki = 330 nM T11072 C5N9GT 11056946 Ki = 650 nM T11072 C0FT4D 11067619 Ki = 1000 nM T11072 C0G3WS 11098166 Ki = 8.5 nM T11072 CK89UG 11101187 Ki = 30 nM T11072 CRU3M5 11110452 Ki = 820 nM T11072 CTBF50 11120893 Ki = 1100 nM T11072 CVE8T3 11121216 Ki = 2 nM T11072 C6CL1Y 11178830 Ki = 100 nM T11072 C9N5QU 11200511 Ki = 29.5 nM T11072 C6D1MZ 11223004 Ki > 1000 nM T11072 C6MI9K 11235335 Ki = 2.512 nM T11072 C90WSG 11248705 Ki = 630.96 nM T11072 CAPX71 11259254 Ki = 5.012 nM T11072 C8JW3Z 11260311 Ki = 45 nM T11072 CO25MT 11270107 Ki = 1.995 nM T11072 C9BLC7 11304596 Ki = 0.1585 nM T11072 CJS9C0 11304851 IC50 > 3200 nM T11072 CTN62X 11328382 Ki = 0.7943 nM T11072 CBV52J 11384146 Ki = 4.7 nM T11072 CF4OX6 11397149 Ki = 0.3162 nM T11072 CGV14H 11402988 Ki = 0.7 nM T11072 CCA2X4 11407766 Ki < 10000 nM T11072 CKL9J7 11419978 Ki = 0.2512 nM T11072 CG4ST6 11464355 Ki = 10 nM T11072 CCGF98 11476072 Ki = 19.95 nM T11072 C6D1MA 11584660 Ki = 199.53 nM T11072 CKWA60 11591924 Ki = 251.19 nM T11072 CGX8F6 11596869 Ki > 2400000 nM T11072 CNEV03 11626724 IC50 = 4 nM T11072 CKO3M0 11647963 IC50 = 0.45 nM T11072 CX7FR8 11655728 Ki = 0.1 nM T11072 C75URP 11668825 IC50 = 0.1 nM T11072 CHK5I2 11712756 Ki = 0.1259 nM T11072 CX9VH0 11720815 Ki = 0.1585 nM T11072 C18COQ 11722647 IC50 = 11 nM T11072 C74LAD 11723305 Ki = 4.6 nM T11072 CZE25U 11725335 Ki = 52 nM T11072 CSL02Y 11726413 Ki = 112 nM T11072 C3T9XB 11727140 Ki = 740 nM T11072 CL97KG 11728004 Ki = 110 nM T11072 CD49YX 11740144 Ki = 0.9 nM T11072 CPZ5N7 11740280 Ki = 2.5 nM T11072 C6B4YJ 11743042 Ki = 26 nM T11072 CYV02C 11747350 Ki = 330 nM T11072 CJ0NV3 11754707 Ki = 3801.89 nM T11072 CG2WS6 11759467 Ki = 420 nM T11072 CK1C4D 11774585 Ki = 7.943 nM T11072 CFQ7B0 11777831 Ki = 340 nM T11072 CJ3G6W 11777940 Ki = 2.5 nM T11072 CB3NF0 11778645 Ki = 35 nM T11072 C9XNZ8 11779840 Ki = 23 nM T11072 CYZP79 11794624 Ki = 199.53 nM T11072 C7EWM8 11794750 EC50 = 1.3 nM T11072 CCR26G 11795333 IC50 = 0.6 nM T11072 C4U5IW 11795525 EC50 = 7.1 nM T11072 CV5UF3 11795644 IC50 = 0.5 nM T11072 CC69IB 11796081 IC50 = 3.2 nM T11072 C6TM2A 11796257 Ki = 12.59 nM T11072 CDJ7T1 11796806 EC50 = 1.5 nM T11072 C7R9MY 11796807 EC50 = 3 nM T11072 C0DTJ5 11796808 EC50 = 11 nM T11072 CAMY96 11797158 Ki = 0.18 nM T11072 CIK15Y 11797562 EC50 = 2.6 nM T11072 C3U7IY 11797644 IC50 = 0.3 nM T11072 CN2BP0 11797998 Ki = 0.11 nM T11072 CY75KM 11797999 Ki = 1.5 nM T11072 CQ35ZC 11798094 EC50 = 0.2 nM T11072 CFMK96 11798502 IC50 = 5.2 nM T11072 C9AT7N 11798621 EC50 = 15 nM T11072 CS19AU 11800592 Ki = 0.11 nM T11072 CQHI29 11808793 Ki = 40 nM T11072 CUI5G6 11809037 Ki = 8 nM T11072 CF9T0I 11810310 Ki = 690 nM T11072 CL1J7U 11822996 Ki = 380 nM T11072 CVW4B5 11824522 Ki = 380 nM T11072 C8JQL7 11957735 IC50 > 10000 nM T11072 C2QAC7 12406830 Ki = 54 nM T11072 CVSW49 12987128 Ki > 10000 nM T11072 CC0ZK7 13096730 Ki = 39 nM T11072 C06OWP 14011045 IC50 = 470 nM T11072 CWK85F 14519865 Ki = 103 nM T11072 C87QBZ 14547414 Ki = 15 nM T11072 CJG80D 14547415 Ki = 228 nM T11072 CYW76P 14742527 Ki > 1000 nM T11072 CC47XA 14973078 Ki = 12 nM T11072 CY4E2W 14977566 Ki = 15 nM T11072 CJ16HE 15011385 IC50 = 220 nM T11072 C7VAI1 15011772 Ki > 10000 nM T11072 CTX2Z7 15233110 IC50 = 13000 nM T11072 CK9Q8B 15340760 Ki = 1.1 nM T11072 CS2G0L 15480709 Ki = 31 nM T11072 C30CHU 15512229 Ki < 316.23 nM T11072 C4R5JF 15516681 IC50 = 1.35 nM T11072 C62NLP 15516682 IC50 = 0.65 nM T11072 CX0P5R 15516683 IC50 = 1.8 nM T11072 C2NJ5B 15521385 IC50 = 0.9 nM T11072 CQ07MV 15521391 IC50 = 0.8 nM T11072 C7Y9LU 15521392 IC50 = 1.2 nM T11072 CO91MH 15549970 Ki = 1.4 nM T11072 C1LWZ6 16006605 Ki = 966 nM T11072 CK36NS 16006607 Ki = 70 nM T11072 C1SR0O 16071847 Ki > 5000 nM T11072 CD3E8L 16093484 Ki = 260 nM T11072 CEW91O 16093485 Ki = 143 nM T11072 CZ1WJ4 16117151 Ki = 410 nM T11072 CM32ZX 16117153 Ki > 5000 nM T11072 CXTB90 16117279 Ki = 1496 nM T11072 C1F2LS 16118795 Ki > 5000 nM T11072 C69VDS 16118923 Ki = 1340 nM T11072 CZ2IS9 16660294 Ki > 10000 nM T11072 C0T9ZY 17947861 Ki = 10 nM T11072 C1X0VH 18007501 Ki = 22 nM T11072 CI4Z6D 18007533 Ki = 32 nM T11072 C5J1AK 18007572 Ki = 5.6 nM T11072 CF6PM0 18007586 Ki = 3.7 nM T11072 C6MFH3 18007589 Ki = 7.3 nM T11072 CHXQ26 18366015 IC50 = 89.13 nM T11072 CUJ1C8 18691541 IC50 = 3.631 nM T11072 CI1DQ5 18691565 IC50 = 100 nM T11072 CP07ZI 18691566 IC50 = 7.079 nM T11072 C7G3UV 18694165 IC50 = 3.981 nM T11072 CIEM47 18694195 IC50 = 10 nM T11072 CZV26X 18694196 IC50 = 1.995 nM T11072 CE5GD1 18975338 IC50 = 1.8 nM T11072 CP8S5X 18975369 IC50 = 0.3 nM T11072 CYJ48A 19066163 Ki = 37 nM T11072 C0BE1M 19066188 Ki = 340 nM T11072 CV5FR6 19066200 Ki = 230 nM T11072 C4RU6O 19066201 Ki = 90 nM T11072 CN96TB 19066203 Ki = 88 nM T11072 C60SWJ 19066205 Ki = 70 nM T11072 C5MS9T 19066235 Ki = 42000 nM T11072 C6AOE8 19426635 IC50 > 1000 nM T11072 CQ3JL0 19956256 IC50 = 478.63 nM T11072 C7T8JC 19958494 Ki > 10000 nM T11072 C6LI5E 19958507 Ki > 10000 nM T11072 CT1C6U 20255884 Ki = 330 nM T11072 CBY03N 20846175 Ki < 10000 nM T11072 CQ17TR 21460878 IC50 = 31.62 nM T11072 C2JT9X 21460905 IC50 = 1.585 nM T11072 C3T5HF 21509921 Ki = 85 nM T11072 CT7XG9 21830793 Ki = 88.3 nM T11072 CBN84K 22065997 Ki > 10000 nM T11072 C2Z0BJ 22326660 Ki = 251.19 nM T11072 CD80PB 22326688 Ki = 1.585 nM T11072 CJ3P6O 22326704 Ki = 2.512 nM T11072 CRU1N2 22611622 Ki = 150 nM T11072 CH5C7X 23288790 Ki = 8.6 nM T11072 CR1F5X 23374587 IC50 = 1.1 nM T11072 C6GBU8 24762221 EC50 = 5.012 nM T11072 CD7CV6 24771120 Ki > 2000 nM T11072 CJ4RO1 24804774 Ki = 1 nM T11072 CK84BF 24804775 EC50 = 1 nM T11072 C1Z3OQ 24804941 Ki = 1.995 nM T11072 C6AE2U 24804942 Ki = 19.95 nM T11072 C1ZYM4 24804943 Ki > 1000 nM T11072 CDC91N 24839550 Ki = 691.83 nM T11072 CF8I9P 24845776 Ki = 1258.93 nM T11072 C93JWY 24865538 Ki = 1 nM T11072 C5F2VL 24865539 Ki = 12.59 nM T11072 CW9N1Z 24865540 Ki = 199.53 nM T11072 C8PXH7 24865541 Ki = 5.012 nM T11072 CN5VB4 24865542 Ki = 1.259 nM T11072 CPF5E2 24865543 Ki = 1.259 nM T11072 CGDV58 24865724 Ki = 1.585 nM T11072 C3HK0J 24865725 Ki = 0.5012 nM T11072 C5TX3M 24865726 Ki = 1.585 nM T11072 C0O6FX 24865727 Ki = 1.585 nM T11072 CER0O4 24881201 Ki = 3.4 nM T11072 C5ZK1C 24881202 Ki = 0.9 nM T11072 C1OF5Z 24881203 Ki = 0.95 nM T11072 C02XDI 24881204 Ki = 1.7 nM T11072 C82DUO 24881264 Ki = 11.3 nM T11072 CIA98Y 24881550 Ki = 24 nM T11072 CMS4W9 24881551 Ki > 1000 nM T11072 CDW36L 24881552 Ki = 219 nM T11072 C8OGB4 24881617 Ki = 0.6 nM T11072 CFMS90 24881618 Ki = 1 nM T11072 CUF79T 24881619 Ki = 13 nM T11072 C18SOA 24881686 Ki = 3.9 nM T11072 CCQY75 24881687 Ki = 151 nM T11072 C49DNT 24881688 Ki > 1000 nM T11072 CJSL82 24881689 Ki = 0.95 nM T11072 CXA24K 24881752 Ki = 0.9 nM T11072 CZ5Q6P 24881753 Ki = 1.4 nM T11072 C4FWN1 24881754 Ki = 2.3 nM T11072 COU24N 24882192 Ki = 79 nM T11072 C43RTZ 24882193 Ki = 0.3 nM T11072 C8B4YF 24882266 Ki = 13 nM T11072 CNO84Q 24882267 Ki = 13 nM T11072 CK6R9A 24882268 Ki = 1.5 nM T11072 C6L7KS 24887518 Ki < 3162.28 nM T11072 CI53SE 24893978 Ki = 140 nM T11072 CYJ5G1 25067564 Ki = 2270 nM T11072 CM2T9Y 25263297 Ki > 2000 nM T11072 CFJM71 25263302 Ki > 2000 nM T11072 CXZH39 44138098 Ki = 0.05012 nM T11072 CUOD42 44138104 Ki = 0.1 nM T11072 CSK83C 44213966 IC50 = 0.3162 nM T11072 C69CVF 44213967 IC50 = 7.943 nM T11072 C34HLC 44213968 IC50 = 0.7943 nM T11072 C92CVD 44214329 Ki = 0.5 nM T11072 CYN83E 44214559 EC50 = 0.2 nM T11072 CIN1S4 44272400 IC50 = 42.66 nM T11072 C13QRS 44272402 IC50 = 776.25 nM T11072 CJ15FQ 44272419 IC50 = 151.36 nM T11072 CC2OD4 44278111 Ki > 10000 nM T11072 CRMA84 44278114 Ki > 10000 nM T11072 CF0Y4M 44278115 Ki > 10000 nM T11072 C08LZS 44279525 Ki = 0.4 nM T11072 C1OI7G 44279549 Ki = 0.5 nM T11072 CFWE96 44279550 Ki = 1.24 nM T11072 C7DR8P 44279889 Ki = 1.71 nM T11072 CDP67Q 44292364 Ki = 0.45 nM T11072 CS3HX6 44292365 Ki = 0.25 nM T11072 C32ARH 44292367 Ki = 3.5 nM T11072 C1Y0JR 44292375 Ki = 0.29 nM T11072 CZL18K 44310169 Ki = 762 nM T11072 C5Q1VH 44311908 Ki > 10000 nM T11072 CYI2D8 44311953 Ki > 5000 nM T11072 CD2TL3 44318323 IC50 = 3.3 nM T11072 CV8WZ0 44318454 IC50 = 302 nM T11072 CXJL56 44318842 IC50 > 1000 nM T11072 C40NAS 44322821 IC50 = 25.12 nM T11072 CZ7JF6 44322823 IC50 = 15.85 nM T11072 CSQT84 44322859 IC50 > 1000 nM T11072 CR0DQ4 44322885 IC50 = 50.12 nM T11072 C5WL1J 44322886 IC50 = 7.943 nM T11072 C37UTX 44322916 IC50 = 158.49 nM T11072 C3C1OY 44322934 IC50 = 3.162 nM T11072 CJC37P 44322940 IC50 > 1000 nM T11072 C2LV3J 44322952 IC50 > 1000 nM T11072 C1MTR2 44322963 IC50 > 1000 nM T11072 C5R2NL 44322965 IC50 > 1000 nM T11072 C5UFN9 44323074 IC50 = 3.162 nM T11072 C3CZF1 44323147 IC50 = 12.59 nM T11072 CEH78W 44323156 IC50 = 39.81 nM T11072 CW7F6I 44323157 IC50 = 125.89 nM T11072 CLN5S4 44323161 IC50 = 63.1 nM T11072 CQI51B 44323162 IC50 = 10 nM T11072 CHG3F0 44323163 IC50 > 1000 nM T11072 CR14CB 44323200 IC50 > 1000 nM T11072 C9LUP6 44323231 IC50 = 10 nM T11072 CD26JI 44323253 IC50 = 5.012 nM T11072 CE7B0T 44323254 IC50 = 6.31 nM T11072 CE8VP0 44323267 IC50 > 1000 nM T11072 C97JUP 44323355 IC50 = 1.4 nM T11072 CS9Z7Q 44323506 IC50 = 12 nM T11072 CS7NA2 44337678 Ki = 2 nM T11072 CU4F3W 44337731 Ki = 240 nM T11072 CUT24A 44338900 Ki = 17 nM T11072 CL2KT5 44339071 Ki = 110 nM T11072 CT8FG6 44339072 Ki = 98 nM T11072 C9AP7L 44341609 IC50 = 1.3 nM T11072 CW2MP5 44341625 IC50 = 11 nM T11072 C5S2NC 44341637 IC50 = 3.2 nM T11072 C0WZJ1 44341657 IC50 = 4.5 nM T11072 CIC09X 44341707 IC50 = 1.2 nM T11072 C8B4XQ 44341783 IC50 = 21 nM T11072 CLD14T 44341798 IC50 = 7.3 nM T11072 CME4B2 44342506 Ki = 0.56 nM T11072 CVI4J5 44342507 Ki = 5.6 nM T11072 CX8LV0 44342508 Ki = 0.45 nM T11072 C3I7YQ 44342518 Ki = 0.38 nM T11072 CAUL48 44342705 Ki = 3 nM T11072 CNSF41 44342722 Ki = 0.45 nM T11072 CIA3M0 44342727 Ki = 0.76 nM T11072 C7OQD9 44342767 Ki = 0.68 nM T11072 CQV5X1 44342783 Ki = 2 nM T11072 CC08TZ 44342784 Ki = 0.38 nM T11072 C9KGS3 44342785 Ki = 0.46 nM T11072 CBGP96 44342823 Ki = 4 nM T11072 C1URA6 44342830 Ki = 0.42 nM T11072 C9K5VL 44342969 Ki = 0.8 nM T11072 C7YS8F 44342993 Ki = 0.7 nM T11072 CPWJ26 44343212 Ki = 1995.26 nM T11072 C9Y8WE 44344504 IC50 = 200 nM T11072 C6N3XK 44345317 IC50 < 1000 nM T11072 C2EHY6 44346844 IC50 = 1200 nM T11072 CX3ZL5 44351656 Ki = 0.74 nM T11072 CUXH48 44352308 Ki = 1620 nM T11072 CVO43T 44358407 Ki = 57 nM T11072 CN2E0L 44362284 IC50 = 110 nM T11072 CS3J6N 44363580 Ki > 100 nM T11072 CVS5L1 44364110 IC50 = 37 nM T11072 C6CJ7S 44373641 EC50 = 0.24 nM T11072 C0AJ1Z 44376262 Ki = 7.8 nM T11072 C6FLR4 44376263 Ki = 6.1 nM T11072 CS32NH 44376272 Ki = 9.5 nM T11072 C9S8OK 44376278 Ki = 29 nM T11072 COT84H 44376280 Ki = 12 nM T11072 C89EPR 44376282 Ki = 12 nM T11072 CHFE56 44376283 Ki = 29 nM T11072 C94ACX 44376362 Ki = 74 nM T11072 C3JEU0 44376363 Ki = 16 nM T11072 C0W7LR 44376383 Ki = 7.4 nM T11072 C86TNU 44376395 Ki = 6.2 nM T11072 CTF4O0 44376491 Ki = 27 nM T11072 CRE24Q 44376492 Ki = 9.3 nM T11072 CKDU28 44376494 Ki = 29 nM T11072 C8C2KA 44376516 Ki = 8.6 nM T11072 CQVX74 44376541 Ki = 8.8 nM T11072 CJ90UO 44376588 Ki = 11 nM T11072 CL7O3J 44376722 Ki = 8.5 nM T11072 C2MAB6 44376723 Ki = 11 nM T11072 C0U9RL 44383728 Ki = 31 nM T11072 C5RYQ7 44383729 Ki = 4.5 nM T11072 CM0T9D 44383737 Ki = 1.8 nM T11072 CV4C3R 44383738 Ki = 8.2 nM T11072 CIS4L0 44394222 Ki = 0.3 nM T11072 CN02LY 44395762 Ki = 2300 nM T11072 C93XHA 44395809 Ki = 210 nM T11072 CTA27N 44395810 Ki = 2300 nM T11072 C9A4NM 44395832 Ki = 140 nM T11072 C4B0OI 44397588 Ki = 158.49 nM T11072 C5FP0R 44397589 Ki = 1258.93 nM T11072 CE3G8U 44397670 Ki = 398.11 nM T11072 C1KA3F 44400359 Ki = 10 nM T11072 C9THQ3 44402868 Ki = 125.89 nM T11072 C1EI5Q 44402869 Ki = 158.49 nM T11072 CV0PC9 44402870 Ki = 12.59 nM T11072 CV15IH 44402871 Ki = 79.43 nM T11072 CD20SO 44402874 Ki = 251.19 nM T11072 CM45GD 44402875 Ki = 251.19 nM T11072 CG1WU9 44402876 Ki = 25.12 nM T11072 C6WNI4 44402877 Ki = 100 nM T11072 CDL1F6 44402878 Ki = 125.89 nM T11072 CLR72M 44402879 Ki = 100 nM T11072 CZL9Y8 44402880 Ki = 199.53 nM T11072 CHU6W5 44402881 Ki = 158.49 nM T11072 C8ZJ7W 44402882 Ki = 50.12 nM T11072 C6M8WP 44402883 Ki = 31.62 nM T11072 CKX16M 44402884 Ki = 25.12 nM T11072 CHG01P 44402885 Ki = 15.85 nM T11072 CD37FS 44402886 Ki = 398.11 nM T11072 CI4MO9 44402887 Ki = 125.89 nM T11072 CX89BK 44402888 Ki = 199.53 nM T11072 CSDV68 44402893 Ki = 501.19 nM T11072 CY4FD0 44402894 Ki = 15.85 nM T11072 CRWN42 44402895 Ki = 251.19 nM T11072 C1B4QL 44403095 Ki = 6.51 nM T11072 C1YL7Z 44403098 Ki = 168.2 nM T11072 CFV98A 44403101 Ki = 209.2 nM T11072 C6OY9S 44403102 Ki = 345.1 nM T11072 CH4SX6 44403105 Ki = 328.7 nM T11072 C12FIH 44403106 Ki = 15.4 nM T11072 CI0WG5 44404225 Ki = 0.5012 nM T11072 C7FAW3 44404229 Ki = 0.7943 nM T11072 C0MXR4 44404230 Ki = 15.85 nM T11072 C7OD6Q 44404236 Ki = 2.512 nM T11072 C5W2KR 44404240 Ki = 0.5012 nM T11072 CI50CY 44404241 Ki = 3.981 nM T11072 CF69DU 44404244 Ki = 7.943 nM T11072 CE0NI6 44404245 Ki = 2.512 nM T11072 CLW3P7 44404249 Ki = 1.259 nM T11072 CF8LN5 44404253 Ki = 2.512 nM T11072 C3LI6E 44404258 Ki = 2.512 nM T11072 C2NH8G 44404260 Ki = 7.943 nM T11072 C7R5HU 44404264 Ki = 7.943 nM T11072 CVTZ13 44404268 Ki = 1 nM T11072 C18ISW 44404272 Ki = 3.162 nM T11072 C4LKC1 44404394 Ki = 34.7 nM T11072 C3EJ4G 44404396 Ki = 103.1 nM T11072 CG87PW 44409290 Ki > 360 nM T11072 CL59HA 44431531 Ki = 56 nM T11072 C6JK5A 44431532 Ki = 7 nM T11072 C5LNH6 44431533 Ki = 88 nM T11072 CLX73C 44431534 Ki = 14 nM T11072 CCV62B 44431535 Ki = 10 nM T11072 C4P5XG 44431536 Ki = 0.9 nM T11072 CYPR70 44431537 Ki = 1 nM T11072 CKZF16 44439165 Ki = 794.33 nM T11072 CA4HZ3 44439167 Ki = 630.96 nM T11072 CT0C4I 44443093 Ki = 0.5012 nM T11072 C8E1AC 44443094 Ki = 1 nM T11072 CZ6BK9 44443095 Ki = 1.995 nM T11072 CV5T2C 44443096 Ki = 3.162 nM T11072 CT1S6L 44443097 Ki = 2.512 nM T11072 CF1V8O 44443098 Ki = 6.31 nM T11072 CHZ48Q 44443101 Ki = 1.995 nM T11072 CQ53TV 44443130 Ki = 0.3981 nM T11072 CEZ6U8 44443131 Ki = 0.5012 nM T11072 CN4XZ6 44443132 Ki = 1.259 nM T11072 CZL97F 44455426 Ki = 706 nM T11072 CYS7T4 44455943 Ki = 1275 nM T11072 C6BFI0 44456033 Ki = 1097.9 nM T11072 CG91RD 44456395 Ki = 1156 nM T11072 C12XGE 44456400 Ki = 684 nM T11072 C5ZML8 44457907 IC50 = 8 nM T11072 CM3IR1 44457909 IC50 = 3.35 nM T11072 CAS01K 44458044 IC50 = 0.83 nM T11072 CGD04W 44458045 IC50 = 20.3 nM T11072 C94DNM 44458229 IC50 = 2.63 nM T11072 CTV0R6 44458239 IC50 = 0.33 nM T11072 CM9YD2 44458486 IC50 = 27.3 nM T11072 C32FOA 44458487 IC50 = 1.98 nM T11072 CP2F5J 44460810 Ki = 20 nM T11072 C6GHE9 44460826 Ki = 40 nM T11072 CXB7G1 44461149 Ki = 63 nM T11072 CZ5E2H 44461168 Ki = 51 nM T11072 C8YD0T 44461234 Ki = 28 nM T11072 CJAI80 44461247 Ki = 74 nM T11072 C3R5WE 44461248 Ki = 40 nM T11072 C9TXL1 44461249 Ki = 8.4 nM T11072 CI0RQ9 44461251 Ki = 130 nM T11072 CQ4S9I 44461266 Ki = 145 nM T11072 CO0ZT7 44461293 Ki = 130 nM T11072 C6UTB1 44461297 Ki = 24 nM T11072 C9GJ3W 44461298 Ki = 28 nM T11072 C2ZH0I 44461300 Ki = 65 nM T11072 CCT61W 44461306 Ki = 31 nM T11072 C09MBT 44461308 Ki = 165 nM T11072 CJHL27 44461335 Ki = 26 nM T11072 CT06WG 44461336 Ki = 122 nM T11072 CB8C2D 44461416 Ki = 71 nM T11072 CIN15X 44461425 Ki = 26 nM T11072 CHL8S2 44461443 Ki = 14 nM T11072 C2IDH4 44461586 Ki = 57 nM T11072 CQ2IX7 44461606 IC50 > 1000 nM T11072 C3D4HR 44537940 Ki > 5000 nM T11072 CJ7U3K 44554227 Ki > 5000 nM T11072 CM0I1P 44554393 Ki > 5000 nM T11072 CNHA47 44554395 Ki = 2761 nM T11072 CB23PH 44560995 Ki = 0.55 nM T11072 CVA67X 44568347 Ki = 2700 nM T11072 CZO5Y8 44580740 Ki = 1.585 nM T11072 C4N6PM 44580741 Ki = 0.5012 nM T11072 C0XVL5 44580783 Ki = 25.12 nM T11072 C4SD7P 44580784 Ki = 0.3162 nM T11072 CNOU35 44581235 Ki = 3.162 nM T11072 CO6E5K 44581260 Ki = 1 nM T11072 CS6HG9 44581603 Ki = 1.259 nM T11072 C1HAQ2 44581604 Ki = 3.981 nM T11072 C5NS6H 44581972 Ki = 416.87 nM T11072 CK8Z1P 44581973 Ki = 741.31 nM T11072 C3UQ9Z 44581974 Ki = 457.09 nM T11072 CRCH48 44582675 Ki = 1062 nM T11072 CEJ4R8 44582676 Ki = 713 nM T11072 CZGP86 44582677 Ki = 3418 nM T11072 C5QB4K 44582678 Ki = 1440 nM T11072 CXL25V 44582706 Ki > 10000 nM T11072 C8MR1X 44582707 Ki = 1835 nM T11072 C4IT1N 44582708 Ki = 1436 nM T11072 C17LZR 44585926 Ki > 1000 nM T11072 CCU63Y 44585927 Ki > 1000 nM T11072 C5PG1H 44585928 Ki > 1000 nM T11072 CY1LE7 44585929 Ki > 1000 nM T11072 CMY8N9 44585945 Ki > 1000 nM T11072 C0S5ER 44585946 Ki > 1000 nM T11072 CSF39B 44588698 Ki = 125.89 nM T11072 C7SKM1 44588720 Ki = 79.43 nM T11072 CI6SO1 44588721 Ki = 7.943 nM T11072 CB14UQ 44588722 Ki = 158.49 nM T11072 CNK64D 44588742 Ki = 251.19 nM T11072 CAT73D 44588743 Ki = 1258.93 nM T11072 C6DK3E 44588744 Ki = 1258.93 nM T11072 C9BO7K 44588745 Ki = 6.31 nM T11072 CD2CU8 44588771 Ki = 1995.26 nM T11072 CDIQ25 44588772 Ki = 251.19 nM T11072 C4EH6O 44592207 Ki = 0.7943 nM T11072 CZ5I1N 44592208 Ki = 5.012 nM T11072 CKM8T7 44592209 Ki = 0.1995 nM T11072 CDJ32U 44592249 Ki = 0.2512 nM T11072 CS2FL4 44592250 Ki = 0.1585 nM T11072 CL17WU 44592251 Ki = 0.3162 nM T11072 CJCL64 44592252 Ki = 0.3981 nM T11072 CM0I3E 44592294 Ki = 0.3981 nM T11072 CQ04EG 44592295 Ki = 1.585 nM T11072 C65XQL 44592296 Ki = 0.07943 nM T11072 CEB2S1 44592297 Ki = 0.3162 nM T11072 CP51QS 44592332 Ki = 3.162 nM T11072 CD2Z4J 44592333 Ki = 0.631 nM T11072 C7NCT2 44592334 Ki = 15.85 nM T11072 CHY20X 44592335 Ki = 3.981 nM T11072 C5H7XK 44592371 Ki = 0.3981 nM T11072 CZ0W1I 44593711 Ki = 251.19 nM T11072 C98UOH 45260312 Ki = 100 nM T11072 C6Y0LZ 45260341 Ki = 630.96 nM T11072 CHLR80 45260355 Ki = 251.19 nM T11072 C31CPA 45260363 Ki = 316.23 nM T11072 CNQ7G1 45260372 Ki = 100 nM T11072 C2YL4K 45260377 Ki = 63.1 nM T11072 C7LRZ1 45260417 Ki = 3981.07 nM T11072 C2MC4K 46881463 EC50 = 501.19 nM T11072 CSQ4C9 46881468 EC50 = 3162.28 nM T11072 C1JSH9 46899637 Ki = 0.01995 nM T11072 C3MSL0 46899638 Ki = 0.1995 nM T11072 CV3LP2 46899639 Ki = 0.1585 nM T11072 CGHZ15 46899640 Ki = 0.1585 nM T11072 CN9FC3 46900150 Ki = 0.1 nM T11072 C40ZJO 46900451 Ki = 0.1259 nM T11072 CNC02A 46900453 Ki = 0.1585 nM T11072 CTCH14 46900455 Ki = 0.1259 nM T11072 CP41AQ 46900457 Ki = 0.1259 nM T11072 CR3L4I 46900459 Ki = 0.1585 nM T11072 CK17PA 46900606 Ki = 0.1259 nM T11072 CQ2K1C 46900608 Ki = 0.1259 nM T11072 C5ZT1B 46900610 Ki = 0.3162 nM T11072 C1NAX4 46900612 Ki = 0.1 nM T11072 CT0SQ2 46900614 Ki = 0.3162 nM T11072 CXD9S3 46900776 Ki = 0.1585 nM T11072 C8I7SJ 46900778 Ki = 1.995 nM T11072 C7QDM9 46900782 Ki = 0.1585 nM T11072 C15FMY 46900954 Ki = 0.03981 nM T11072 C8W1FU 46900956 Ki = 0.1 nM T11072 CH35BV 46900958 Ki = 0.1585 nM T11072 CO69SV 46905266 Ki = 25 nM T11072 C2LZJ0 49783209 Ki = 1304 nM T11072 C57SMG 49783415 Ki = 5686 nM T11072 C0TG6I 49783419 Ki = 2856 nM T11072 C4HIZ8 49799868 Ki = 15 nM T11072 C3OHN0 49850566 Ki = 0.5012 nM T11072 C4R2YS 49850567 Ki = 0.1995 nM T11072 CSGQ38 49850568 Ki = 0.3981 nM T11072 C8P5KH 49850569 Ki = 0.2512 nM T11072 C07JTU 49850570 Ki = 0.1585 nM T11072 C6FP9W 49850571 Ki = 0.1585 nM T11072 C3BVK5 49850668 Ki = 0.2512 nM T11072 C6P3RH 49850669 Ki = 0.1995 nM T11072 CGYT84 49850670 Ki = 0.631 nM T11072 C6Y3DW 49850671 Ki = 0.5012 nM T11072 CK68QR 49850672 Ki = 0.2512 nM T11072 CI6O9A 49850673 Ki = 0.1259 nM T11072 COFA76 49850768 Ki = 0.3162 nM T11072 C4IX5R 49850769 Ki = 0.3162 nM T11072 CXLT59 49850770 Ki = 0.2512 nM T11072 C48DOX 49850771 Ki = 1.585 nM T11072 CN5XR1 49850772 Ki = 0.1585 nM T11072 CR4EZ0 49850870 Ki = 0.1259 nM T11072 C5K4EC 49850872 Ki = 0.2512 nM T11072 C8AW0R 49850874 Ki = 0.3162 nM T11072 CB2K6D 49850877 Ki = 0.3162 nM T11072 C85KPE 49850980 Ki = 0.3981 nM T11072 C5U3YD 49850982 Ki = 0.631 nM T11072 CV62IZ 49850984 Ki = 0.1585 nM T11072 CED9V6 49852000 Ki = 0.631 nM T11072 CA0PW5 49852001 Ki = 0.1995 nM T11072 C5S6BY 49852002 Ki = 0.1585 nM T11072 C13ZTD 49852003 Ki = 0.3162 nM T11072 CK17IE 49852105 Ki = 0.5012 nM T11072 C2RY0J 50878551 Ki = 100 nM T11072 C1W6TV 50898777 Ki = 3162.28 nM T11072 CXMZ73 50898778 Ki > 10000 nM T11072 C67IRJ 50908804 Ki = 0.5012 nM T11072 CLOB24 50908805 Ki = 39.81 nM T11072 CE4KP1 51050257 Ki > 10000 nM T11072 CX9AF4 52942551 Ki = 0.1 nM T11072 CR0G5U 52942644 Ki = 0.1259 nM T11072 CCF97B 52943811 Ki = 2.512 nM T11072 C2FG9O 52943861 Ki = 0.3981 nM T11072 C9G4CI 52943891 Ki = 2.512 nM T11072 CCVP06 52944840 Ki = 5.012 nM T11072 CJ49MX 52946290 Ki = 3.981 nM T11072 CK5ER0 52947414 Ki = 0.07943 nM T11072 CAVB03 52947615 Ki = 0.1259 nM T11072 C1HRK4 52947622 Ki = 1.259 nM T11072 C4ZC1K 52948697 Ki = 1.995 nM T11072 CPA2G4 52951481 Ki > 10000 nM T11072 CYP0I3 52951482 Ki > 10000 nM T11072 C32YWL 53324045 Ki = 628 nM T11072 CRQF15 53325242 Ki = 844 nM T11072 CG24AT 53381002 Ki > 10000 nM T11072 C8WHT5 56593934 Ki = 10000 nM T11072 CW89BT 56595402 Ki > 1000 nM T11072 C4C3XQ 56595529 Ki > 1000 nM T11072 C6W1RA 56649648 Ki = 122 nM T11072 C2SW7J 56649649 Ki = 361 nM T11072 CQTR49 56649650 Ki = 92 nM T11072 CH37LU 56663451 IC50 > 10000 nM T11072 CCY98O 56935645 Ki = 44 nM T11072 C1TC7Q 56963799 Ki = 5237 nM T11072 C1LEH8 67268994 Ki = 2112 nM T11072 CLS9Y8 67650695 IC50 = 5 nM T11072 C63DCO 67650716 IC50 = 13 nM T11072 CP9V6A 69836292 Ki = 251.19 nM T11072 CQH61C 70681318 Ki = 63 nM T11072 CT38JR 70683414 Ki = 157 nM T11072 CPO08R 70691861 Ki > 1500 nM T11072 CD37EI 70691866 Ki = 6.7 nM T11072 C3XNC2 71450247 Ki = 2360 nM T11072 C8P9EA 71450983 IC50 = 9.3 nM T11072 C2ZGV6 71452688 Ki = 250 nM T11072 CAQF34 71455625 Ki > 10000 nM T11072 CMJ1O9 71457409 Ki > 10000 nM T11072 CPO82B 71458050 Ki = 31.62 nM T11072 CS83IF 71459269 Ki > 10000 nM T11072 CG0WO9 71459954 Ki = 65 nM T11072 CJT49M 71459969 IC50 = 2.1 nM T11072 C63YLA 71461049 Ki = 2569 nM T11072 CJD96I 71461050 Ki > 10000 nM T11072 C6VL5X 71461632 Ki = 0.55 nM T11072 C85EAM 71461714 IC50 = 13 nM T11072 C4P3JU 71462776 Ki > 10000 nM T11072 C3GUQ2 71462777 Ki > 10000 nM T11072 C8Z0NM 72550642 Ki = 418 nM T11072 CL6W2Q 72550645 Ki = 122 nM T11072 C78LYM 72698087 Ki > 10000 nM T11072 C63HPK 72698088 Ki > 10000 nM T11072 CC6Q5R 72771081 Ki < 100 nM T11072 CC65OA 73213195 Ki = 28.84 nM T11072 CW83DK 73213196 Ki = 625 nM T11072 CCV91B 73346042 Ki = 234.6 nM T11072 C2E7QW 75201901 Ki = 9300 nM T11072 C8IDL3 75306277 Ki = 63.1 nM T11072 C4P8QN 76312087 Ki = 225.2 nM T11072 C3A8EB 76312089 Ki = 5463 nM T11072 COM84H 76315630 Ki = 599.4 nM T11072 CR0XQ1 76319309 Ki = 1124 nM T11072 CU6YO0 76322954 Ki = 2034 nM T11072 CP3YB5 76322955 Ki = 5404 nM T11072 C3IPW2 76322957 Ki = 393.2 nM T11072 CDY2S1 76326510 Ki = 1238 nM T11072 C6LUP2 76326511 Ki > 10000 nM T11072 C2Z5SX 76326513 Ki = 6288 nM T11072 CNU59S 76326515 Ki = 1491 nM T11072 C5HJ9N 76330154 Ki = 975.4 nM T11072 C1XTC0 76330155 Ki = 3817 nM T11072 C9SX2Q 76330156 Ki = 2874 nM T11072 C5KHL8 76330158 Ki = 7788 nM T11072 CEMZ15 118464420 Ki = 2904 nM T11072 CV2L6O 118464425 Ki = 3830 nM T11072 CFNG86 118464427 Ki > 10000 nM T11072 C7ODW3 122195524 Ki > 900 nM T11072 C3VDY7 122197403 Ki = 14 nM T11072 C1MFJ3 122197404 Ki = 67 nM T11072 C7GO0U 122197405 Ki = 1.8 nM T11072 CLW53P 122483274 Ki = 1404 nM T11072 CO63ET 122483280 Ki = 462 nM T11072 C4QM2E 124247485 Ki = 636 nM T11072 CTBN56 127026052 Ki = 758.58 nM T11072 CBE56W 127026514 Ki = 1280 nM T11072 C0SZI4 127026515 Ki = 28 nM T11072 CQ0ZT9 127035062 Ki = 451 nM T11072 CU49VE 127036186 Ki = 398.11 nM T11072 CG06BD 127036932 Ki = 213.8 nM T11072 CVW71O 127036953 Ki = 125.89 nM T11072 C50GOC 130442480 Ki = 8100 nM T11072 CM04RF 130442572 Ki = 8900 nM T11072 CAVB41 132584404 Ki > 10000 nM T11072 CBU81N 134149168 Ki > 10000 nM T11072 C6N8GM 135367405 Ki = 165 nM T11072 C6LU0C 135367816 Ki > 10000 nM T11072 CD2TH9 135367820 Ki > 10000 nM T11072 C5AMD9 135367857 Ki = 147 nM T11072 CGBW93 135410312 Ki = 9.333 nM T11072 CVE08Y 135458392 Ki = 1457 nM T11072 CP7HN4 135458393 Ki = 1367 nM T11072 CS8XJ6 135458394 Ki = 454 nM T11072 C9B7XA 135458410 Ki = 630 nM T11072 CFV9A3 135458427 Ki = 82 nM T11072 CKX4N8 135458428 Ki = 747 nM T11072 C7DF4S 135464159 Ki = 288.4 nM T11072 CP9XN7 135500023 Ki < 100000 nM T11072 C6I9RK 135516645 Ki = 1778.28 nM T11072 CQI23C 135516796 Ki = 870.96 nM T11072 C3FV9I 135527031 Ki = 263.03 nM T11072 CA1M8B 135966709 Ki = 160 nM T11072 CUKO20 136020617 Ki > 10000 nM T11072 COF0U5 136020618 Ki > 10 nM T11072 CF89JI 136030596 Ki > 10000 nM T11072 CE8GB9 136030693 Ki > 10000 nM T11072 C65VFI 136030744 Ki > 10000 nM T11072 COIX80 136054961 Ki > 10000 nM T11072 C19GLK 136116062 Ki > 10000 nM T11072 CS0JL5 136118616 Ki > 10000 nM T11072 C5UDW3 136118620 Ki = 6835 nM T11072 C8I6UN 136118621 Ki > 10000 nM T11072 CD7OE2 136118652 Ki > 10000 nM T11072 C0W1TM 136118658 Ki = 2552 nM T11072 C42FCS 136118661 Ki = 8867 nM T11072 CB12QP 136152964 Ki = 1437.4 nM T11072 CFX06E 136152966 Ki = 1810 nM T11072 C37YXA 136152971 Ki = 233 nM T11072 CY0C1X 136152972 Ki > 10000 nM T11072 CSNE17 136179514 Ki = 588.84 nM T11072 CAE39V 136188797 Ki > 10000 nM T11072 CLAP52 136259032 Ki > 10000 nM T11072 C7KC3T 145963830 Ki = 2200 nM T11072 CHDN35 145964150 Ki = 9700 nM T11072 C1KH2E 145964159 Ki = 2000 nM T11072 C12OVL 145965034 Ki > 10000 nM T11072 C5W4LM 145965940 Ki > 10000 nM T11072 C81VUO 145967771 Ki > 10 nM T11072 CJS56K 145967795 Ki = 8600 nM T11072 CQJ5O8 145971635 Ki > 10000 nM T11072 C7BVC1 145972374 Ki = 3300 nM T11072 C79TNE 145972796 Ki = 8500 nM T11072 C6XIN0 145974114 Ki > 10000 nM T11072 CD8ZL6 145974750 Ki > 10 nM T11072 C6PH4F 145975226 Ki = 530 nM T11072 C71CYU 145975946 Ki > 10000 nM T11072 C2TN8W 145976085 Ki = 800 nM T11072 C6BFY7 145977338 Ki = 1900 nM T11072 C0Y6QO 145977799 Ki = 1600 nM T11072 C3BI1R 145978113 Ki = 5300 nM T11072 CQU8R0 145978665 Ki = 2700 nM T11072 C6AV9G 145978819 Ki > 10000 nM T11072 C87MSW 145980271 Ki = 1074 nM T11072 C8I7QL 145980875 Ki = 4431 nM T11072 CNJH37 145986752 Ki = 10000 nM T11072 CUGO10 145988693 Ki = 752 nM T11072 C4GV8Q 145990586 Ki = 857 nM T11072 CC2G1V 146025727 Ki = 4100 nM T11072 C6P3SR 153287553 Ki > 10000 nM T11072 CV9G7Z 153287572 Ki > 10000 nM T11072 CO85KL 153287574 Ki > 10000 nM T11072 CUSA24 155519891 Ki > 10000 nM T11072 CB79ZW 155536080 Ki > 10000 nM T11072 C3N9VU 10251906 Ki > 500 nM T11072 D00CRA 1574 Ki = 1220 nM T11072 D00FHZ 124007 IC50 = 2200 nM T11072 D00OBS 44559159 Ki > 10000 nM T11072 D01HRV 9847194 EC50 = 0.8 nM T11072 D01KAX 135453290 Ki = 7870 nM T11072 D02EPZ 24782016 Ki = 2210 nM T11072 D02UWB 1809 IC50 = 3.388 nM T11072 D03DET 10287730 Ki = 0.7943 nM T11072 D03KPA 15870567 Ki = 45 nM T11072 D03MVY 10198700 Ki = 1.7 nM T11072 D03TDN 1342 Ki = 6.18 nM T11072 D03XAE 10775128 Ki = 16 nM T11072 D03ZHB 44455973 Ki > 10000 nM T11072 D04AQE 1833 Ki = 4.1 nM T11072 D04AZE 3277600 Ki < 10000 nM T11072 D04DLR 128018 Ki = 700 nM T11072 D04TPO 16006492 Ki = 1272 nM T11072 D05GDP 599482 Ki > 10000 nM T11072 D05XGR 6918647 Ki = 251.19 nM T11072 D07LRJ 5312149 Ki = 251.19 nM T11072 D08CKM 9863250 Ki = 3162.28 nM T11072 D08DOG 25130235 Ki = 120 nM T11072 D08OFG 11177588 Ki > 10000 nM T11072 D08VGJ 9904281 Ki = 1265 nM T11072 D09AVG 11831220 Ki = 39.6 nM T11072 D09HJL 10331436 Ki > 10000 nM T11072 D09OYA 2107 Ki = 150 nM T11072 D09PIN 3378093 Ki = 260 nM T11072 D09RPR 16737207 Ki > 10000 nM T11072 D09WIL 10028436 Ki = 25.12 nM T11072 D0C3EX 1797 Ki = 16 nM T11072 D0C5GF 6918515 Ki = 6225 nM T11072 D0C5XQ 1832 Ki = 20 nM T11072 D0CK9K 6918513 Ki = 290 nM T11072 D0D8GV 9830741 Ki > 500 nM T11072 D0D9YW 3292447 Ki = 31.62 nM T11072 D0F6CD 5202 Ki = 0.5 nM T11072 D0H7PC 6918553 Ki > 3981.07 nM T11072 D0H9QG 5312148 Ki = 3162.28 nM T11072 D0K9MT 10912152 Ki = 5.3 nM T11072 D0KQ9H 10468938 EC50 = 2.3 nM T11072 D0KS0I 24894910 EC50 > 10000 nM T11072 D0L5MW 181743 Ki = 49 nM T11072 D0M7SY 9910352 Ki = 100 nM T11072 D0O3GF 1220 Ki = 115 nM T11072 D0P4KF 44269078 Ki = 105 nM T11072 D0PN8D 44351692 Ki = 0.7 nM T11072 D0QM3E 9870500 Ki = 1 nM T11072 D0R3GW 10296414 Ki = 1.585 nM T11072 D0V5HV 4296 IC50 = 610 nM T11072 D0V7OO 10386282 IC50 = 0.6 nM T11072 D0XX2U 16006606 Ki = 446 nM T11072 D0Y9TL 13702393 Ki = 3594 nM T89636 D03VOJ 8768 IC50 = 239000 nM T89636 C54JUR 25043 IC50 = 141000 nM T89636 C70HVL 77888 IC50 = 137000 nM T89636 CPI2E4 80447 IC50 = 71600 nM T89636 C07AKH 786691 IC50 = 20000 nM T89636 CY4MC6 3505109 IC50 = 145000 nM T89636 CGN9J7 44267478 IC50 = 25000 nM T89636 CH4Q6A 145964401 IC50 = 6100 nM T89636 CHU61S 145964420 IC50 = 600 nM T89636 C6YCA8 145964710 IC50 = 700 nM T89636 CV6F7L 145966788 IC50 = 600 nM T89636 CBWX17 145967285 IC50 = 900 nM T89636 COR9X3 145972736 IC50 = 700 nM T89636 CQ0M2X 145972809 IC50 = 7500 nM T89636 CF95RZ 145972878 IC50 = 600 nM T89636 CXI0D1 145975081 IC50 = 700 nM T89636 CG84ZR 145975487 IC50 = 400 nM T89636 C91FOT 145976006 IC50 = 800 nM T89636 C3F4UH 145978039 IC50 = 500 nM T37505 CGL7H5 51348369 EC50 > 10000 nM T37505 CY6E1X 51348522 EC50 = 93 nM T37505 C6DM5O 51348672 EC50 = 3.5 nM T37505 C9ZUM4 51348956 EC50 = 15 nM T37505 CO1TP5 51354469 EC50 = 270 nM T37505 CN6KF4 51354470 EC50 > 10000 nM T37505 C8BD6Z 51355032 EC50 = 29 nM T37505 C12HEA 51355324 EC50 = 144.54 nM T37505 CZ0BL8 51355598 EC50 = 810 nM T37505 CL7MC9 51355880 EC50 = 90 nM T37505 C0RG6P 51356141 EC50 = 91 nM T37505 C30TOB 51356430 EC50 = 110 nM T37505 C4AT0S 58466401 EC50 = 110 nM T37505 C7RLI4 67438968 EC50 = 190 nM T37505 CHS21O 69925894 EC50 = 487 nM T37505 C10TPN 86658399 EC50 = 134 nM T37505 CQ1B3I 118727604 EC50 = 4.7 nM T37505 CYP27W 118727605 EC50 = 1.1 nM T37505 CCWI47 118727606 EC50 = 0.68 nM T37505 CYM3V1 118727607 EC50 = 0.57 nM T37505 CF0BE6 118727608 EC50 = 1.4 nM T37505 CDF7M6 118727609 EC50 = 11 nM T37505 CP76TC 118727610 EC50 = 10 nM T37505 CSIT80 118727611 EC50 = 3 nM T37505 C7OT9H 118727612 EC50 = 2 nM T37505 CU2L4D 118727613 EC50 = 5.1 nM T37505 C90KRT 118727614 EC50 = 4.7 nM T37505 CLWC51 118727615 EC50 = 6.6 nM T37505 COIJ51 118727616 EC50 = 2.5 nM T37505 CH1S0U 118727617 EC50 = 4300 nM T37505 CEXT05 118727618 EC50 = 2200 nM T37505 CJ4V7M 118727619 EC50 > 25000 nM T37505 C42HGL 118727620 EC50 > 25000 nM T37505 CXB81W 118727621 EC50 = 3000 nM T37505 C0BKC9 118727622 EC50 = 600 nM T37505 C8MER1 118727623 EC50 = 560 nM T37505 CMJ0D4 118727624 EC50 = 650 nM T37505 CD4SM9 118727625 EC50 = 1200 nM T37505 CHVP35 118727626 EC50 > 25000 nM T37505 CRC5S8 118727627 EC50 = 1600 nM T37505 CHI6W3 118727628 EC50 > 25000 nM T37505 CQXT04 118727629 EC50 = 770 nM T37505 CG7HA5 118727630 EC50 = 960 nM T37505 CVGN49 118727631 EC50 = 720 nM T37505 C9Y8WD 118727632 EC50 = 1300 nM T37505 C8N4HA 118727633 EC50 = 11000 nM T37505 C7WO9I 118727634 EC50 = 130 nM T37505 COEY28 118727635 EC50 = 1500 nM T37505 C7S1KZ 118727636 EC50 = 1500 nM T37505 C20LNY 118727637 EC50 = 130 nM T37505 CYE7S5 118727638 EC50 = 19000 nM T37505 CATF34 118727639 EC50 = 210 nM T37505 C02HDB 118727640 EC50 = 360 nM T37505 CQI21J 118727641 EC50 = 450 nM T37505 C02YRT 118727642 EC50 = 580 nM T37505 CO8UA6 118727643 EC50 = 730 nM T37505 CO8Q3S 118727644 EC50 = 1300 nM T37505 CDT86V 118727645 EC50 = 3600 nM T37505 CDY1I4 118727646 EC50 = 1500 nM T37505 C9FI1L 118727647 EC50 = 23000 nM T37505 CIL9J3 118727648 EC50 = 6200 nM T37505 CJU6X2 118727649 EC50 = 10000 nM T37505 C0REY5 118727650 EC50 = 13000 nM T37505 CIT21Z 118727651 EC50 = 1200 nM T37505 C3S7JO 118727652 EC50 = 1500 nM T37505 CF3P7I 118727653 EC50 = 2000 nM T37505 C1D8KH 118727654 EC50 = 1200 nM T37505 C2BW3P 118727655 EC50 = 2100 nM T37505 CW03IV 118727656 EC50 = 1200 nM T37505 C9RF0N 118727657 EC50 = 360 nM T37505 C54RMV 118727658 EC50 = 1200 nM T37505 CKU52W 118727659 EC50 = 3400 nM T37505 CNW1I2 118727660 EC50 = 330 nM T37505 CF8QH1 118727661 EC50 = 1100 nM T37505 CLA6W1 118727662 EC50 = 3200 nM T37505 C37MAL 118727663 EC50 = 900 nM T37505 C4RPF7 118727664 EC50 = 2100 nM T37505 C48BRL 118727665 EC50 = 1600 nM T37505 C4FVE6 118727666 EC50 = 670 nM T37505 CXE79D 118727667 EC50 = 4500 nM T37505 C0UXA7 118727668 EC50 = 640 nM T37505 C7RUQ1 118727669 EC50 = 3800 nM T37505 CS3VH7 118727670 EC50 = 230 nM T37505 CH6I1F 118727671 EC50 = 44 nM T37505 C6C5PN 118727672 EC50 = 61 nM T37505 C79EHP 118727673 EC50 = 750 nM T37505 C3ILN2 118727674 EC50 = 340 nM T37505 CG1HJ2 118727675 EC50 = 72 nM T37505 CGE42T 118727676 EC50 = 90 nM T37505 CAO47J 118727677 EC50 = 120 nM T37505 CN9S3M 118727678 EC50 = 94 nM T37505 C7PS1R 118727679 EC50 = 170 nM T37505 CLY0D3 118727680 EC50 = 35 nM T37505 CIB24M 118727681 EC50 = 280 nM T37505 CRB5S3 118727682 EC50 = 1100 nM T37505 CE68UZ 118727683 EC50 = 66 nM T37505 CBA72G 118727684 EC50 = 110 nM T37505 CO6E3R 118727685 EC50 = 260 nM T37505 CW61GT 118727686 EC50 = 980 nM T37505 CX3T8O 118727687 EC50 = 320 nM T37505 CAN96J 118727688 EC50 = 1200 nM T37505 CA2XT0 118727689 EC50 = 5500 nM T37505 C8AOB1 118727690 EC50 = 460 nM T37505 C6JS5L 118727691 EC50 = 6400 nM T37505 CZ7F9Y 118727692 EC50 > 30000 nM T37505 CG08ZK 118727693 EC50 = 1200 nM T37505 C1D9MT 118729996 EC50 = 6000 nM T37505 C1IL7Q 118729997 EC50 = 500 nM T37505 CU32MX 118729998 EC50 > 10000 nM T37505 CV3B9G 118729999 EC50 > 10000 nM T37505 CWXK69 118730000 EC50 > 10000 nM T37505 CBC3A2 118730001 EC50 = 110 nM T37505 CB8P1O 118730002 EC50 = 730 nM T37505 C5HRK2 118730003 EC50 = 170 nM T37505 C4PFH9 118730004 EC50 = 120 nM T37505 CXR69F 118730005 EC50 = 860 nM T37505 CZ6O2M 118730006 EC50 = 1500 nM T37505 CT0B9O 118730007 EC50 = 570 nM T37505 C2O1ZF 118730008 EC50 = 160 nM T37505 CO6JX4 118730009 EC50 = 460 nM T37505 C5KO2V 118730010 EC50 = 190 nM T37505 CZ1WR2 118730011 EC50 = 170 nM T37505 CHCV20 118730012 EC50 = 260 nM T37505 CE69SA 118730013 EC50 = 410 nM T37505 CXVW90 118730014 EC50 = 690 nM T37505 CD1SL4 118730015 EC50 > 270000 nM T37505 CE87VL 118730016 EC50 > 81000 nM T37505 CD8EC0 118730017 EC50 > 110000 nM T37505 CYX4N6 118730018 EC50 = 2500 nM T37505 C1S0FP 118730161 EC50 = 880 nM T37505 CHL7B3 118730162 EC50 = 1.2 nM T37505 CN96AV 118730163 EC50 > 100 nM T37505 C3LXM0 118730164 EC50 = 1.8 nM T37505 C5PI2B 118730165 EC50 = 2 nM T37505 C4Z0SK 118730166 EC50 = 5.8 nM T37505 C4PL5S 118730167 EC50 = 1.4 nM T37505 CGO38U 118730168 EC50 = 1.7 nM T37505 CWV2G1 118730169 EC50 = 0.66 nM T37505 CA82GD 134129964 EC50 = 583 nM T37505 C67XEO 134130076 EC50 = 9549.93 nM T37505 C30XQY 134130159 EC50 > 10000 nM T37505 CS1HG2 134130337 EC50 = 537.03 nM T37505 CM2KL8 134130378 EC50 = 414 nM T37505 CP46CD 134130396 EC50 = 345 nM T37505 C9ZA2N 134130466 EC50 = 616 nM T37505 CUV60C 134130479 EC50 = 3890.45 nM T37505 C1GF8C 134130714 EC50 > 10000 nM T37505 CQH75P 134130956 EC50 = 5860 nM T37505 CJ85HT 134131000 EC50 > 10000 nM T37505 CKSH98 134131406 EC50 = 7870 nM T37505 C4XIW6 134131464 EC50 = 2630 nM T37505 CCZ97L 134131577 EC50 = 3700 nM T37505 CWC9G4 134131592 EC50 = 1440 nM T37505 C48SIG 137628671 EC50 = 25 nM T37505 CH7D3Q 155510728 EC50 = 125.89 nM T37505 C4ZF7S 155516531 EC50 = 158 nM T37505 C6L9GA 155524121 EC50 = 316 nM T37505 CL0QH7 155524265 EC50 = 125.89 nM T37505 CG7S5N 155524317 EC50 = 398 nM T37505 CX71YN 155525986 EC50 = 96 nM T37505 CZR67H 155530522 EC50 = 501 nM T37505 CQ2ZC6 155538983 EC50 = 501 nM T37505 C16GNF 155555151 EC50 = 125.89 nM T37505 CMDG07 155561859 EC50 = 63 nM T37505 CDA8R4 155566459 EC50 = 1258.93 nM T37505 D0O6ZN 58466521 EC50 = 3.1 nM T40474 D03ZBT 11626560 IC50 = 0.51 nM T40474 D04LVK 57379345 IC50 = 271 nM T40474 D07POC 176870 IC50 > 12500 nM T40474 D0IQ6P 25102847 IC50 = 1.3 nM T40474 D0K8KX 5280343 IC50 = 580 nM T40474 D0R0MW 5329102 IC50 = 2000 nM T40474 D0U3SY 49806720 IC50 > 5000 nM T40474 D0W5HK 216239 IC50 = 5750 nM T40474 D00DRL 44137946 IC50 = 0.4 nM T40474 D01GFX 11640390 IC50 > 12500 nM T40474 D01LCC 17754438 EC50 = 0.3 nM T40474 D02RJY 11442891 IC50 > 10000 nM T40474 D02UFQ 11620908 IC50 = 4200 nM T40474 D03HUX 49792852 IC50 > 10000 nM T40474 D03LWG 53235510 IC50 = 3011 nM T40474 D05OMT 45142457 IC50 = 0.6 nM T40474 D06EGV 44603533 IC50 = 4.7 nM T40474 D07ARN 25182860 IC50 = 4 nM T40474 D07EHV 44814409 IC50 > 10000 nM T40474 D07HPJ 11476171 IC50 > 10000 nM T40474 D07OJZ 25145656 IC50 = 0.13 nM T40474 D08FDX 24901704 IC50 = 12 nM T40474 D09ETH 16118392 IC50 = 14 nM T40474 D0D1GF 42642645 IC50 = 0.4 nM T40474 D0E3TC 44259 IC50 = 69.2 nM T40474 D0FA6S 54576299 IC50 = 2.7 nM T40474 D0G0BL 44181686 IC50 = 1 nM T40474 D0KX7I 56960363 IC50 = 0.74 nM T40474 D0L9PA 56960447 IC50 = 0.69 nM T40474 D0LW0T 68289010 IC50 = 1.995 nM T40474 D0O0LS 25141092 IC50 > 10000 nM T40474 D0O6WV 24794418 IC50 < 2.512 nM T40474 D0OK2N 24864821 IC50 = 9 nM T40474 D0P1CV 46191454 IC50 > 10000 nM T40474 D0P6DJ 151194 IC50 > 10000 nM T40474 D0Q9UX 16718576 IC50 > 10000 nM T40474 D0R8QG 25171648 IC50 < 1 nM T40474 D0U2BH 65064 Ki = 3300 nM T40474 D0YT8P 46911863 IC50 = 0.95 nM T40474 D0ZI1F 11494412 Ki = 355 nM T40474 D0ZU5F 24779724 IC50 = 3.1 nM T40474 D03BNU 59604787 IC50 > 3500 nM T40474 D0LF0O 135441202 IC50 = 3990 nM T40474 D09HEV 6539952 IC50 > 20000 nM T40474 D0T3ME 156422 IC50 > 30000 nM T40474 CM20CY 10393 IC50 > 20000 nM T40474 C63WLY 89644 IC50 > 10 ug.mL-1 T40474 C5JE2Z 104860 IC50 = 7 ug.mL-1 T40474 CNIW58 107905 IC50 = 10000 nM T40474 CI1NA5 159926 IC50 = 4.3 ug.mL-1 T40474 CYBA43 177458 IC50 = 4.3 ug.mL-1 T40474 CDZ65K 199472 IC50 = 10000 nM T40474 C1UAQ4 342168 IC50 > 100000 nM T40474 CW72UL 388108 IC50 = 6660 nM T40474 CK0L4O 442514 IC50 = 400 nM T40474 C1ZG2U 449087 IC50 > 10000 nM T40474 CL68XJ 598695 IC50 = 4300 nM T40474 C86GHK 759814 IC50 = 7630 nM T40474 CE56TK 823838 IC50 = 12300 nM T40474 CJIQ30 1010856 IC50 = 1300 nM T40474 CT73CE 1014283 IC50 = 15800 nM T40474 CD5FI0 1048794 IC50 = 3500 nM T40474 C8KVJ3 1048795 IC50 = 2200 nM T40474 C5V3DJ 1048811 IC50 = 8100 nM T40474 CFCV05 1212526 IC50 = 10300 nM T40474 CY0EX9 2226536 IC50 > 100000 nM T40474 C8F6DW 2716301 IC50 > 100000 nM T40474 CNZO64 2716309 IC50 > 100000 nM T40474 C31KAP 2743369 IC50 = 113 nM T40474 CRHC32 2933553 IC50 = 675 nM T40474 CHPQ17 3327252 IC50 = 28300 nM T40474 C0Z5WX 3699929 IC50 = 3700 nM T40474 C73RMN 4067150 IC50 = 43000 nM T40474 C0LY1H 4269048 IC50 = 69000 nM T40474 C9NMI6 4938134 IC50 = 5870 nM T40474 C4NF9V 5095151 IC50 = 5680 nM T40474 C8IAR2 5281657 IC50 > 100000 nM T40474 CI68PW 5283685 IC50 = 71500 nM T40474 CXK0S6 5283727 IC50 = 78000 nM T40474 CZIU69 5304328 IC50 > 100000 nM T40474 CDQ3M7 5359485 IC50 = 5.4 ug.mL-1 T40474 C54BYP 5360741 IC50 > 10 ug.mL-1 T40474 CDK3J0 5703619 IC50 = 109 nM T40474 C0KTW5 6441913 IC50 > 20000 nM T40474 CUPQ08 6539985 IC50 > 50000 nM T40474 CMEZ23 6540005 IC50 > 50000 nM T40474 CQR03O 7117329 IC50 > 100000 nM T40474 C7L8RJ 9506623 IC50 = 11190 nM T40474 C4G9WR 9547398 IC50 > 100000 nM T40474 C76CUP 9547698 IC50 = 47600 nM T40474 C59FOQ 9658158 IC50 = 780 nM T40474 C1E2DV 9826083 IC50 > 10000 nM T40474 CM5Z8X 9869943 IC50 > 100000 nM T40474 C5YF4Z 9870238 Ki = 1 nM T40474 C12PKF 9871380 IC50 > 10000 nM T40474 CPQ13K 9933545 IC50 > 20000000 nM T40474 C26QHZ 10005638 IC50 > 10000 nM T40474 CR8DA1 10024683 IC50 > 100000 nM T40474 CLA93G 10047202 IC50 = 27500 nM T40474 C3LCH5 10047545 IC50 > 100000 nM T40474 C7YD1X 10048045 IC50 > 25000 nM T40474 CUJR40 10062694 EC50 > 2000 nM T40474 C7L2MG 10100985 IC50 = 7770 nM T40474 CREM37 10151881 IC50 = 3900 nM T40474 C59FGN 10165455 IC50 > 1000 nM T40474 CC78NE 10179293 IC50 = 2110 nM T40474 CEW30I 10217590 IC50 = 6500 nM T40474 CSGD16 10246246 IC50 > 7000 nM T40474 CVZ03W 10254297 Ki = 2450 nM T40474 CJGH26 10275985 IC50 = 8990 nM T40474 C3FL9K 10295633 IC50 = 1500 nM T40474 C7SFI1 10296883 IC50 > 10000 nM T40474 CA8B5T 10390073 IC50 > 10000 nM T40474 CN61JB 10392099 Ki = 460 nM T40474 CO1I5Q 10415576 IC50 = 170 nM T40474 C4CP7K 10423452 IC50 = 4400 nM T40474 C4KTX2 10428645 Ki = 3830 nM T40474 C7HBP6 10429593 IC50 > 10000 nM T40474 CP9XE8 10686611 IC50 > 100000 nM T40474 C83QWV 10714343 IC50 = 3120 nM T40474 C0KD7L 10805173 IC50 > 100000 nM T40474 COEU74 11151773 IC50 = 1790 nM T40474 CV18ED 11204241 IC50 = 22 nM T40474 C8G5WP 11210533 IC50 = 1120 nM T40474 C8T2NG 11211389 IC50 = 7400 nM T40474 CT3K9Z 11213588 IC50 = 350 nM T40474 C1R5QA 11219056 IC50 = 830 nM T40474 CQ4XT3 11224593 IC50 = 6700 nM T40474 C2W5RC 11235063 IC50 > 50000 nM T40474 CB95CD 11243660 IC50 = 50 nM T40474 CG93PJ 11259074 IC50 = 1000 nM T40474 CBOP58 11293798 Ki > 10000 nM T40474 CNP57I 11305951 IC50 = 17 nM T40474 C4VAE6 11310709 IC50 = 56 nM T40474 CLX54H 11317348 IC50 > 10000 nM T40474 C87KQR 11324313 IC50 = 4 nM T40474 C0W4CU 11324689 IC50 = 7 nM T40474 CGP80V 11328586 IC50 = 650 nM T40474 C4RHB6 11340470 Ki = 3 nM T40474 CL2VR4 11342673 IC50 = 4 nM T40474 CSG09F 11347373 IC50 = 150 nM T40474 C1G8SZ 11347754 IC50 = 220 nM T40474 CEC31B 11351900 IC50 = 370 nM T40474 C26BZX 11362471 Ki > 10000 nM T40474 CB45PJ 11362483 IC50 = 20000 nM T40474 C9B4XP 11363872 IC50 = 230 nM T40474 CP4ZO0 11375301 IC50 = 300 nM T40474 C27LKY 11381132 IC50 = 6 nM T40474 C4IH5E 11383525 IC50 = 20000 nM T40474 CD68KH 11387226 IC50 = 40 nM T40474 CWXB93 11397177 Ki > 10000 nM T40474 CT3VP7 11398307 IC50 = 3320 nM T40474 C5K9DA 11419123 IC50 = 170 nM T40474 C73PUW 11420344 IC50 = 460 nM T40474 CFJ6B2 11441375 IC50 = 20000 nM T40474 CGB80I 11450766 IC50 = 1150 nM T40474 CYSV74 11451912 IC50 = 45 nM T40474 C4Q7XD 11474276 IC50 = 6900 nM T40474 C2Z7WP 11486459 IC50 = 20000 nM T40474 CH1WJ0 11497322 IC50 = 90 nM T40474 C6XN2I 11504713 IC50 = 1.5 nM T40474 CGB1U0 11504995 IC50 = 70 nM T40474 CWYR62 11510244 IC50 = 1000 nM T40474 C3UPR5 11510560 Ki = 50 nM T40474 CAYS74 11517264 IC50 = 8000 nM T40474 CH2IZ9 11517688 IC50 = 1500 nM T40474 CIQR82 11518616 IC50 = 65 nM T40474 C98ENG 11525727 Ki = 2 nM T40474 CL7X4Q 11530963 IC50 = 35000 nM T40474 C3WJZ0 11533908 IC50 = 114 nM T40474 CTG83F 11539329 Ki > 2900 nM T40474 C8Y2BI 11540273 IC50 = 132 nM T40474 C0QY6X 11540508 IC50 = 80 nM T40474 C20ZUM 11540724 IC50 = 48 nM T40474 C1KAT5 11546617 IC50 = 780 nM T40474 C4I6AF 11555216 IC50 = 160 nM T40474 CK7QU2 11555957 IC50 = 130 nM T40474 C41ASL 11560856 IC50 = 110 nM T40474 CACS26 11561968 Ki > 2000 nM T40474 CZW01X 11568819 IC50 = 10000 nM T40474 CQ3BT9 11575401 Ki = 35.2 nM T40474 C7TH0B 11576617 IC50 = 40.6 nM T40474 CJ01BI 11577131 IC50 = 5200 nM T40474 CJ1OR3 11582499 IC50 = 6600 nM T40474 CUK13J 11583264 IC50 = 6400 nM T40474 C0NWH1 11584471 IC50 = 150 nM T40474 CMIL86 11590363 Ki > 2900 nM T40474 C6XLM1 11591094 IC50 = 80 nM T40474 CDIW70 11597571 IC50 = 18.3 nM T40474 C6C9WI 11598848 IC50 = 28 nM T40474 CFPB69 11599241 IC50 = 125 nM T40474 C69FYK 11604142 Ki = 130 nM T40474 CD61EN 11604265 IC50 = 9640 nM T40474 CI95OG 11611059 IC50 = 10000 nM T40474 CV8EU0 11612136 Ki = 38.3 nM T40474 CSA61M 11612145 IC50 = 500 nM T40474 CQ59BR 11613348 IC50 = 510 nM T40474 C5B3XJ 11620410 IC50 = 13700 nM T40474 C5OEV6 11620642 IC50 = 140 nM T40474 CYS46T 11625675 IC50 = 35.6 nM T40474 CN3QM0 11626442 IC50 = 1000 nM T40474 C7QRE8 11627441 IC50 = 260 nM T40474 C3EJ0G 11634384 IC50 = 430 nM T40474 C9T6SC 11640926 Ki > 2900 nM T40474 C9LOW0 11642366 IC50 = 30 nM T40474 CDPI27 11647759 IC50 = 45.3 nM T40474 CK8VJ4 11647760 Ki = 26 nM T40474 CAC63W 11648548 IC50 = 30 nM T40474 C2A9EU 11654090 Ki = 230 nM T40474 CDVJ79 11654729 IC50 = 5000 nM T40474 CH6R1E 11655658 IC50 = 500 nM T40474 C9HK8A 11656580 Ki = 59.7 nM T40474 CSZK05 11662380 Ki = 14 nM T40474 CYFX19 11667754 Ki = 348 nM T40474 C3D2ZQ 11670702 IC50 = 190 nM T40474 CALI63 11671030 IC50 = 54 nM T40474 C2MVE1 11678254 IC50 = 40 nM T40474 CU0E8O 11690457 Ki > 4000 nM T40474 C5VPR3 11696310 IC50 = 2640 nM T40474 C61SMG 11697050 IC50 = 230 nM T40474 CSD2T8 11697436 IC50 = 140 nM T40474 CH18YG 11699504 IC50 = 40 nM T40474 C68QNX 11699573 IC50 = 90 nM T40474 CP2TW6 11703607 IC50 = 760 nM T40474 CB0AP2 11705863 Ki > 4000 nM T40474 C0OWS4 11713310 IC50 = 2 nM T40474 CVPY27 11713579 IC50 = 30 nM T40474 C42VOT 11717068 IC50 = 7000 nM T40474 C6ZR2P 11719648 IC50 = 2800 nM T40474 C45EWD 11723489 IC50 > 7000 nM T40474 C4QX7D 11738454 IC50 = 160 nM T40474 CS5QL4 11749561 IC50 = 20000 nM T40474 CV64JS 11750694 IC50 = 20000 nM T40474 CS78BX 11771327 IC50 = 13 nM T40474 CS36BH 11843159 IC50 = 2400 nM T40474 C9JT4S 11847343 IC50 > 10000 nM T40474 CI7DT1 11857432 IC50 = 39 nM T40474 CBT94Q 11857507 Ki = 201 nM T40474 CCRA82 11857874 IC50 = 107 nM T40474 CET19P 11857948 IC50 = 12 nM T40474 CEA7I9 11857949 IC50 = 14 nM T40474 CT6FE1 11858025 IC50 = 38 nM T40474 C8Q7IX 11858027 Ki = 14 nM T40474 C4M9EV 11858028 IC50 = 45 nM T40474 CWF6K8 11858029 IC50 = 29 nM T40474 CHR92S 11858109 IC50 = 4.9 nM T40474 CB42LX 11858111 IC50 = 136 nM T40474 C7G4EV 11858191 IC50 = 4.9 nM T40474 CTP89H 11858284 IC50 = 9.2 nM T40474 CDKH57 11858286 IC50 = 17 nM T40474 CQ3T1L 11858367 IC50 = 21 nM T40474 CKVS05 11858368 IC50 = 9.6 nM T40474 CVM84A 11858369 IC50 = 33 nM T40474 CX59JL 11858434 IC50 = 72 nM T40474 C8NF6H 11947782 Ki = 1.4 nM T40474 CO8QR4 11962890 Ki = 53.5 nM T40474 C0HE1D 11962891 Ki = 15.8 nM T40474 CFP7M5 11962976 Ki = 0.8 nM T40474 CP89KY 11962977 Ki = 0.8 nM T40474 CCY4J2 11962978 Ki = 2.4 nM T40474 C3XWU1 11963015 Ki = 3.9 nM T40474 CA7Y5P 11963057 Ki = 0.4 nM T40474 CTC31Z 11963059 Ki = 1 nM T40474 C3H4PA 11963103 Ki = 0.9 nM T40474 CI7G5W 11963258 Ki = 1.4 nM T40474 CT1RA7 11963259 Ki = 29 nM T40474 CY8GD6 11963300 Ki = 1.5 nM T40474 CQ2WD1 11963302 Ki = 2.3 nM T40474 CGCX39 11963344 Ki = 0.6 nM T40474 C4O3UR 11963386 Ki = 0.6 nM T40474 CPG89E 11963387 Ki = 1.2 nM T40474 CF3W2N 11963388 Ki = 1.1 nM T40474 CQT2I1 11963389 Ki = 0.7 nM T40474 CT91NG 11963423 Ki = 0.7 nM T40474 CH2A1C 11963425 Ki = 1.2 nM T40474 C1WBC7 11963465 Ki > 20000 nM T40474 CAI8B7 12581296 Ki > 10000 nM T40474 C87DIW 12758175 IC50 > 100000 nM T40474 CDGF78 15282555 IC50 = 1100 nM T40474 CH8VT9 15980822 IC50 = 380 nM T40474 CKTY30 15980908 IC50 = 1100 nM T40474 C3W8ZL 15981007 IC50 = 31 nM T40474 CFY53O 15981074 IC50 = 10 nM T40474 CM2V3O 15981105 IC50 = 46 nM T40474 C7DB2O 15981106 IC50 = 9000 nM T40474 C7QAM2 15981107 IC50 = 30 nM T40474 C3GEP1 15981108 IC50 = 74 nM T40474 CX2YN3 15981109 IC50 = 170 nM T40474 CL5YM4 15981110 IC50 = 5300 nM T40474 CF36EH 15981111 IC50 = 180 nM T40474 CSXI73 15981140 IC50 = 5500 nM T40474 C8UZE2 15981179 IC50 = 14 nM T40474 C8VYW0 15981180 IC50 = 4 nM T40474 CFPW41 16007116 Ki > 2800 nM T40474 CWV9N7 16035631 IC50 = 1000 nM T40474 CQ29YC 16035632 IC50 = 32 nM T40474 C6DEI5 16035634 IC50 = 46 nM T40474 CA9LE6 16036535 IC50 = 0.7 nM T40474 CU0S5T 16040363 IC50 = 25 nM T40474 CK4LA5 16040525 IC50 = 27 nM T40474 C5K3RO 16040526 IC50 = 100 nM T40474 C9C3AE 16040527 IC50 = 26 nM T40474 CYXZ47 16040697 IC50 = 34 nM T40474 CC68WU 16040698 IC50 = 28 nM T40474 CI0U9N 16040699 IC50 = 26 nM T40474 CYT5V7 16040870 IC50 = 25 nM T40474 CTG84Q 16041065 IC50 = 1000 nM T40474 C93MID 16041066 IC50 = 31 nM T40474 CX1SD5 16041234 IC50 = 590 nM T40474 CWC7B6 16041238 IC50 = 33 nM T40474 CE9ZW5 16041961 IC50 = 26 nM T40474 CD85IU 16041962 IC50 = 32 nM T40474 CEDC74 16042706 IC50 = 28 nM T40474 CMB30J 16042707 IC50 = 4 nM T40474 C8NME0 16042894 IC50 = 38 nM T40474 CZI2H3 16043068 IC50 = 150 nM T40474 CZK8V6 16043304 IC50 = 1100 nM T40474 CQG45C 16109001 IC50 = 25000 nM T40474 C1U8XW 16109036 IC50 > 6700 nM T40474 CC0Z4V 16119626 IC50 = 20200 nM T40474 CBC26E 16122938 IC50 = 150 nM T40474 C5VPH9 16129448 IC50 = 5910 nM T40474 CM8H6W 16221866 IC50 = 9 nM T40474 CS15QH 16221868 IC50 = 9 nM T40474 C5J4IM 16221977 IC50 = 120 nM T40474 CL9JZ7 16222081 IC50 = 22 nM T40474 CEJ8X1 16222087 IC50 = 69 nM T40474 C5HEZ9 16222089 IC50 = 55 nM T40474 C2UV9Y 16222392 IC50 = 4 nM T40474 C6VD9W 16223006 IC50 = 270 nM T40474 CVZK29 16223008 IC50 = 7 nM T40474 CX03LD 16223106 IC50 = 8 nM T40474 CJV61A 16223108 IC50 = 11 nM T40474 C2JD4R 16223110 IC50 = 3500 nM T40474 CH72TP 16223116 IC50 = 6 nM T40474 CIKP98 16223215 IC50 = 24 nM T40474 C63SCI 16223221 IC50 = 9 nM T40474 CY9X6O 16223223 IC50 = 34 nM T40474 CWX69H 16223313 IC50 = 190 nM T40474 CA8K5T 16223315 IC50 = 18 nM T40474 C3GCV7 16223402 IC50 = 13 nM T40474 C01MOK 16260214 IC50 = 30000 nM T40474 CXUO14 16457485 IC50 = 79 nM T40474 CPZ65H 16717966 IC50 = 22 nM T40474 CEG90Z 16725054 Ki = 1020 nM T40474 CDW83C 16734139 IC50 = 90 nM T40474 CXM7O6 16734411 IC50 = 78 nM T40474 CR2OZ8 16736063 IC50 = 2 nM T40474 CU5Q9B 16757524 IC50 = 2.7 nM T40474 C9MNP2 17549086 IC50 > 50000 nM T40474 CL9BQ6 17748275 IC50 = 25000 nM T40474 CL4KF7 17748441 IC50 = 35 nM T40474 CED9B3 21081469 IC50 = 2 nM T40474 CI12XN 21081471 IC50 = 19 nM T40474 CR5M9T 21081472 IC50 = 11 nM T40474 CG5T7S 21081475 IC50 = 4 nM T40474 CU38QR 21081477 IC50 = 2 nM T40474 CLX4B2 21081480 IC50 = 900 nM T40474 CD81BA 21081481 IC50 = 860 nM T40474 CHE12T 21081484 IC50 = 50 nM T40474 CFUP56 21081488 IC50 = 990 nM T40474 C5D7CP 21081489 IC50 = 410 nM T40474 CVTB30 21081490 IC50 = 150 nM T40474 CF0E5U 21081500 IC50 = 44 nM T40474 CUIX06 21081503 IC50 = 11 nM T40474 C4D8YP 21081514 IC50 = 180 nM T40474 CAP2Z4 21081515 IC50 = 1400 nM T40474 CH73SG 21081519 IC50 = 440 nM T40474 C7P6KC 21081520 IC50 = 1000 nM T40474 CH4B5K 21081523 IC50 = 45 nM T40474 CC7DW5 21081576 IC50 = 90 nM T40474 C0RW1U 21081728 IC50 = 5 nM T40474 CD6UG2 21081760 IC50 = 8.2 nM T40474 C25UKC 21081761 IC50 = 1.8 nM T40474 CWP90R 21081766 IC50 = 30 nM T40474 C6LK3S 21081770 IC50 = 1.9 nM T40474 CIW7K0 21081771 IC50 = 10 nM T40474 CG1N9F 21081772 IC50 = 70 nM T40474 C2H4AO 21081778 IC50 = 470 nM T40474 C35UXH 21081792 IC50 = 30 nM T40474 CL0H6J 21081793 IC50 = 70 nM T40474 CX7P0G 21110756 IC50 = 62.4 nM T40474 C8DZ3Q 21110757 IC50 = 43.8 nM T40474 CFKZ31 21110871 Ki = 75 nM T40474 CT3DR9 21110879 Ki = 41.1 nM T40474 CXJU48 21110914 Ki = 260 nM T40474 CB1Y2R 21111219 Ki = 35 nM T40474 CH4NS9 21111337 Ki = 7580 nM T40474 C26CBO 21111396 IC50 = 7120 nM T40474 C4Y5ZI 21111478 Ki = 6560 nM T40474 C70WJN 23153333 IC50 = 100 nM T40474 C6JV7W 23400934 IC50 > 7000 nM T40474 CD5S7O 23401001 IC50 > 7000 nM T40474 CF6LO5 23652906 Ki = 1.7 nM T40474 CH2QT3 23653618 IC50 = 2294 nM T40474 CV83NR 24178428 IC50 = 800 nM T40474 C2RV3U 24180608 IC50 > 30000 nM T40474 CA3I4T 24753787 IC50 > 50000 nM T40474 CHU49V 24757938 IC50 = 450 nM T40474 C7YG1N 24759534 IC50 = 1400 nM T40474 CAJ4T2 24762205 IC50 > 10000 nM T40474 CQNP54 24764449 Ki = 0.5 nM T40474 CCPS81 24764502 IC50 > 35000 nM T40474 C2UOE0 24766030 IC50 > 50000 nM T40474 C4Z9CN 24769780 Ki = 3.4 nM T40474 CN8R5S 24779728 IC50 = 6 nM T40474 CO9Z0H 24822598 IC50 = 5300 nM T40474 C51IZL 24822599 IC50 = 3200 nM T40474 CA90EF 24822600 IC50 = 20000 nM T40474 C4A6LB 24823090 IC50 = 5000 nM T40474 C2B4JP 24823091 IC50 = 11000 nM T40474 CF6M3W 24823093 IC50 = 20000 nM T40474 C0NLO8 24823094 IC50 = 20000 nM T40474 C7D8PC 24823095 IC50 = 20000 nM T40474 C14FLQ 24823250 IC50 = 20000 nM T40474 C36BFD 24823252 IC50 = 20000 nM T40474 CBF60S 24823253 IC50 = 20000 nM T40474 CDT3L2 24824050 IC50 = 410 nM T40474 CLN48F 24824051 IC50 = 1100 nM T40474 C0NXE2 24824052 IC50 = 1400 nM T40474 CWTI12 24824188 IC50 = 1600 nM T40474 CQ1A8W 24824189 IC50 = 260 nM T40474 C8RE5C 24824190 IC50 > 4000 nM T40474 C3K1FM 24824191 IC50 > 4000 nM T40474 CV0S5L 24824318 IC50 = 290 nM T40474 CUK14T 24824319 IC50 > 4000 nM T40474 CZ09ID 24824320 IC50 > 4000 nM T40474 CM28KX 24824321 IC50 = 1200 nM T40474 CD57UN 24824322 IC50 = 500 nM T40474 CNI50G 24824323 IC50 = 210 nM T40474 C84VZK 24824448 IC50 = 7600 nM T40474 C5BA7V 24824452 IC50 = 160 nM T40474 CR49SP 24824453 IC50 > 4000 nM T40474 CG64EL 24824454 IC50 > 4000 nM T40474 C0CHG3 24824705 IC50 = 4 nM T40474 C1GX6O 24830124 IC50 = 500 nM T40474 C37CYH 24830125 IC50 = 3400 nM T40474 C7I4WE 24830764 IC50 = 5300 nM T40474 CKZQ07 24851730 IC50 = 1 nM T40474 CE40IJ 24851953 Ki = 1 nM T40474 C2EOB4 24851954 Ki = 7 nM T40474 CMQ4Z1 24864822 IC50 = 12 nM T40474 CI7LE9 24864823 IC50 = 7 nM T40474 CA9K0C 24864824 IC50 = 67 nM T40474 CH6TG1 24864825 IC50 = 26 nM T40474 CY2HJ0 24864993 IC50 = 7 nM T40474 C6T2DF 24864994 IC50 = 6 nM T40474 CEX30T 24865175 IC50 = 3 nM T40474 CN08BH 24871821 Ki = 16 nM T40474 C20VHK 24871823 IC50 = 6 nM T40474 C2QVN9 24871946 Ki = 14.9 nM T40474 CUW72Q 24871947 Ki = 7 nM T40474 CUJ53D 24872065 Ki = 8 nM T40474 CFK2B9 24882503 IC50 > 10000 nM T40474 C43HWQ 24883287 IC50 > 10000 nM T40474 C8DA5Q 24883334 IC50 > 10000 nM T40474 CRZ57M 24886446 Ki > 30000 nM T40474 CBU9V6 24886674 IC50 = 400 nM T40474 CB5TP8 24894992 IC50 = 29000 nM T40474 CFW40U 24894997 IC50 = 45000 nM T40474 CN13JF 24899915 IC50 = 7.6 ug.mL-1 T40474 CBWR97 24899916 IC50 = 1.7 ug.mL-1 T40474 C9F2JD 24899917 IC50 > 10 ug.mL-1 T40474 C64MTI 24900160 IC50 = 2.5 ug.mL-1 T40474 CO2I6Q 24900161 IC50 = 9.4 ug.mL-1 T40474 C4XZ9O 24901679 IC50 = 1000 nM T40474 CQ0E6R 24901680 IC50 = 1000 nM T40474 CNV1L6 24901681 IC50 = 1000 nM T40474 CP82XK 24901682 IC50 = 2.8 nM T40474 CUBK56 24901683 IC50 = 3.1 nM T40474 C7D1LN 24901684 IC50 = 3.8 nM T40474 C3MEZ4 24901685 IC50 = 3.4 nM T40474 CXE2T7 24901686 IC50 = 5 nM T40474 CZD9W5 24901687 IC50 = 2.3 nM T40474 CSU5V3 24901688 IC50 = 1400 nM T40474 CC06QZ 24901689 IC50 = 1.3 nM T40474 CMQ01W 24901690 IC50 = 1.8 nM T40474 CD08VO 24901691 Ki = 1 nM T40474 C0NCI3 24901692 Ki = 7.9 nM T40474 C59ICM 24901693 IC50 = 1 nM T40474 C9WD7I 24901694 Ki = 1.1 nM T40474 C9KJD4 24901695 IC50 = 1.3 nM T40474 C3QKW8 24901696 IC50 = 120 nM T40474 C6NC2G 24901697 IC50 = 610 nM T40474 C7OMW1 24901698 IC50 = 2100 nM T40474 C6UXO8 24901699 IC50 = 116 nM T40474 C34BSE 24901700 IC50 = 130 nM T40474 C2CD9F 24901701 IC50 = 130 nM T40474 CN9W4J 24901702 IC50 = 113 nM T40474 CVAC46 24901703 IC50 = 193 nM T40474 CNK14W 24901705 IC50 = 52 nM T40474 CAN86I 24901706 IC50 = 35 nM T40474 C58CHD 24901707 IC50 = 24 nM T40474 C0UM9A 24901708 IC50 = 69 nM T40474 CSCB80 24901709 IC50 = 20 nM T40474 C6PDE3 24901710 IC50 = 52 nM T40474 C2KI4J 24901711 IC50 = 181 nM T40474 C2UWO4 24901712 IC50 = 60 nM T40474 CF0KV6 24901713 IC50 = 70 nM T40474 CJO43A 24901714 IC50 = 49 nM T40474 C6OAM7 24901715 IC50 = 74 nM T40474 CIH4C8 24901716 IC50 = 63 nM T40474 C15BZP 24949852 IC50 = 360 nM T40474 CZHE50 24949856 IC50 = 760 nM T40474 CLZ23U 24951610 IC50 > 30000 nM T40474 CK0TP9 24964818 Ki = 13 nM T40474 CY8F9A 24965169 Ki = 24 nM T40474 CW7V4J 24965874 Ki = 44 nM T40474 C5W2PG 24965937 Ki = 13.7 nM T40474 C4BD3N 24965938 IC50 = 40 nM T40474 C3DFE7 24966287 IC50 = 600 nM T40474 CZ9A2F 24966649 IC50 = 20 nM T40474 C9JB2R 24966651 IC50 = 910 nM T40474 C4RGC1 24967005 IC50 = 680 nM T40474 CTDN38 24967006 IC50 = 50 nM T40474 CV9DN5 24967007 IC50 = 50 nM T40474 CN4E9Y 24967008 IC50 = 40 nM T40474 CFC75N 24971366 IC50 = 30 nM T40474 C06NYJ 24971367 IC50 = 71 nM T40474 CFI12X 24971368 IC50 = 52 nM T40474 C69UJG 24971369 IC50 = 368 nM T40474 C4EG8R 24993189 IC50 > 10000 nM T40474 CS3Q8B 24995659 Ki > 4000 nM T40474 CMPD60 25012550 IC50 = 3 nM T40474 CUV63L 25013520 IC50 = 98 nM T40474 CRGT98 25013521 IC50 = 163 nM T40474 C7UT3S 25013522 IC50 = 45 nM T40474 C6E2OK 25013523 IC50 = 52 nM T40474 C4RD2A 25013686 IC50 = 1 nM T40474 CDZ0A1 25013841 IC50 = 6 nM T40474 CLP8M2 25013847 IC50 = 4950 nM T40474 CSR31L 25014027 IC50 = 42 nM T40474 CYM8V9 25014029 IC50 = 8 nM T40474 CC1OW5 25014237 IC50 = 3 nM T40474 C6N7KR 25032700 IC50 = 430 nM T40474 CS0P4K 25054599 IC50 = 2000 nM T40474 C2F1YJ 25054600 IC50 = 700 nM T40474 C0UDM4 25054601 IC50 = 90 nM T40474 C8CA3Y 25054857 IC50 = 150 nM T40474 CDYM40 25055101 IC50 = 12 nM T40474 CMH4W3 25055102 IC50 = 70 nM T40474 CQZ95L 25055103 IC50 = 80 nM T40474 C8UGB1 25055104 IC50 = 60 nM T40474 CAE17C 25055344 IC50 = 180 nM T40474 CF7S1D 25064072 IC50 = 1366 nM T40474 C37HTN 25064073 IC50 > 6667 nM T40474 C9B0FR 25064510 IC50 = 104 nM T40474 C6SZR4 25064730 IC50 = 14 nM T40474 CID6R3 25065131 IC50 = 236 nM T40474 CLN3G1 25066842 IC50 = 29 nM T40474 C2KY1G 25094210 IC50 > 10000 nM T40474 C2P0EV 25102846 IC50 = 21.9 nM T40474 C2Y3AV 25113181 IC50 = 900 nM T40474 C6BWZ8 25145145 IC50 > 100 nM T40474 C78YWA 25145716 IC50 > 500 nM T40474 CP9LZ8 25157323 IC50 = 7 nM T40474 C7DML3 25172983 IC50 = 5.7 nM T40474 C85KCS 25178328 IC50 = 6700 nM T40474 CIG4H0 25178539 IC50 = 3300 nM T40474 C4GI6J 25178540 IC50 = 7400 nM T40474 CRF36L 25182856 IC50 = 10 nM T40474 CF39AL 25182859 IC50 = 29 nM T40474 C2W7QI 25183021 IC50 = 25 nM T40474 CM8OT2 25183023 IC50 = 318 nM T40474 C35EQD 25195745 IC50 = 5 nM T40474 CVT64C 25196402 IC50 = 5 nM T40474 C7BO9Q 25196404 IC50 = 3 nM T40474 C9TE8R 25196406 IC50 = 4 nM T40474 C6FGQ1 25206346 IC50 > 10000 nM T40474 CNG96H 25210579 IC50 > 10000 nM T40474 CF8KU4 25212175 IC50 = 17 nM T40474 C84NZM 25218737 IC50 = 4.5 nM T40474 CSB8X6 25218738 IC50 = 5.9 nM T40474 CCE06R 25218739 IC50 = 3.8 nM T40474 C49KED 25218740 IC50 = 2.7 nM T40474 C1VX8J 25218741 IC50 = 3.4 nM T40474 CDGF43 25218742 IC50 = 1 nM T40474 C6HB0N 25218743 IC50 = 3.4 nM T40474 CUN19O 25218744 IC50 = 1 nM T40474 CD4Y3K 25218745 IC50 = 3.2 nM T40474 C1F7CA 25218746 IC50 = 2.6 nM T40474 CYP6O7 25229537 IC50 = 82 nM T40474 CTK56B 25245053 IC50 > 20000 nM T40474 C4AR9G 25268137 IC50 = 30 nM T40474 C4NE9M 42598432 IC50 = 3 nM T40474 CC4VZ1 42598657 IC50 = 13 nM T40474 C6AM3I 42598658 IC50 = 3 nM T40474 CTQ8I9 42599146 IC50 = 10 nM T40474 C23TME 42601406 IC50 = 40 nM T40474 CUN7O3 42604837 IC50 = 31 nM T40474 CU9E4P 42629114 IC50 > 10000 nM T40474 CJ5U1X 42639664 IC50 = 6.4 ug.mL-1 T40474 CTR6H3 44120806 IC50 = 3310 nM T40474 CAK0F2 44155856 IC50 = 1.7 nM T40474 CC1P5L 44156965 IC50 = 25 nM T40474 CE3OF9 44160137 IC50 = 80 nM T40474 CLW80F 44160269 IC50 = 34000 nM T40474 CSH3D6 44177697 IC50 > 5000 nM T40474 C65VUH 44177803 IC50 > 5000 nM T40474 CP68KL 44179965 IC50 = 580 nM T40474 CV71DM 44179999 IC50 = 1 nM T40474 CHF7Y5 44180001 IC50 = 2 nM T40474 CY83ER 44180127 IC50 = 3 nM T40474 CN9T8B 44180247 IC50 = 8 nM T40474 CT19OY 44180935 IC50 = 6 nM T40474 C2L0GB 44181041 IC50 = 6 nM T40474 CJ7UC6 44181042 IC50 = 780 nM T40474 CTC28H 44181146 IC50 = 60 nM T40474 C7RHW9 44181147 IC50 = 51 nM T40474 CJT15D 44181148 IC50 = 2 nM T40474 CJ4W9G 44181149 IC50 = 12 nM T40474 C9S7VY 44181153 IC50 = 0.77 nM T40474 C05TQH 44181355 IC50 = 3 nM T40474 CSB92W 44181357 IC50 = 9 nM T40474 CZ5WA9 44181358 IC50 = 2 nM T40474 CQMU31 44181460 IC50 = 15 nM T40474 CZC1W4 44181461 IC50 = 8 nM T40474 CNJ3Y1 44181654 IC50 = 26 nM T40474 C0PB1K 44181655 IC50 = 280 nM T40474 C9X5RS 44181688 IC50 = 7 nM T40474 C5LOC6 44189142 IC50 = 9 nM T40474 CLY4S0 44194115 IC50 = 47 nM T40474 CT2S5G 44206063 IC50 = 14 nM T40474 C8KNA3 44219632 Ki > 4000 nM T40474 C0VIX4 44219633 Ki > 4000 nM T40474 CF9UB1 44219665 IC50 > 40000 nM T40474 CXPN30 44219666 IC50 > 40000 nM T40474 CVEU45 44219667 IC50 = 9700 nM T40474 CK73NR 44219749 IC50 > 50000 nM T40474 CEL61X 44229839 IC50 = 1800 nM T40474 C73CBF 44247727 IC50 = 32 nM T40474 CNX68G 44256051 IC50 > 10000 nM T40474 CC0EM6 44256053 IC50 = 53 nM T40474 CF8U5T 44256167 IC50 = 160 nM T40474 CWK6F0 44256275 IC50 = 540 nM T40474 C1QXF2 44256314 IC50 = 410 nM T40474 C7NB5X 44256371 IC50 = 56 nM T40474 CV1X8T 44256373 IC50 = 14 nM T40474 CYO29J 44256408 IC50 = 22 nM T40474 CF6SL7 44256410 IC50 = 19 nM T40474 C0B8JY 44256411 IC50 = 2100 nM T40474 CVET85 44256439 IC50 > 10000 nM T40474 CX2I6P 44256441 IC50 = 1700 nM T40474 C1Z2DH 44256477 IC50 > 10000 nM T40474 C0IJ9C 44256478 IC50 > 10000 nM T40474 C0KD4U 44346053 IC50 > 10000 nM T40474 C7KZV2 44414322 IC50 > 50000 nM T40474 CJM06T 44414347 IC50 > 50000 nM T40474 CA98KR 44432441 IC50 > 10000 nM T40474 C4Y8XV 44446930 IC50 > 1000 nM T40474 CWBV18 44446940 IC50 > 1000 nM T40474 CPR51F 44446941 IC50 = 170 nM T40474 CQW9Z1 44447640 IC50 = 40 nM T40474 C32FHX 44447643 IC50 > 2000 nM T40474 CB3V9R 44447645 IC50 = 440 nM T40474 C0RDZ2 44447646 IC50 = 190 nM T40474 CW2FH0 44447647 IC50 = 37 nM T40474 CJM1U2 44473400 IC50 = 0.6 nM T40474 C2XLG0 44512602 IC50 = 612 nM T40474 CD12FA 44512610 IC50 = 1 nM T40474 CG2AV9 44512611 IC50 = 3 nM T40474 C1NJ8A 44512616 IC50 = 7 nM T40474 CLZR72 44512932 IC50 = 2 nM T40474 C6BS4F 44512934 IC50 = 3 nM T40474 CSN2P3 44512937 IC50 = 2 nM T40474 CS0L3K 44512939 IC50 = 1 nM T40474 CVAE31 44512942 IC50 = 17 nM T40474 C74CNZ 44513256 IC50 = 102 nM T40474 CUL04P 44513257 IC50 = 14 nM T40474 CWKE23 44513258 IC50 = 12 nM T40474 CR1P8B 44513259 IC50 = 2 nM T40474 CIG7R6 44513261 IC50 = 1 nM T40474 CUT5I7 44517769 IC50 = 11 nM T40474 CYH6P3 44520205 IC50 > 10000 nM T40474 C4WRN5 44541014 IC50 = 50000 nM T40474 C3VRO9 44557921 IC50 > 10000 nM T40474 C18LQG 44564591 IC50 = 300 nM T40474 C9LZT0 44564592 IC50 = 67 nM T40474 CD2CQ0 44564593 IC50 = 23 nM T40474 C3I0CK 44564664 IC50 = 320 nM T40474 CUSN60 44564665 IC50 = 21 nM T40474 CH7OL6 44564666 IC50 = 24 nM T40474 CU3G5Z 44564667 IC50 = 250 nM T40474 C0N2OH 44564668 IC50 = 16 nM T40474 CPRU17 44564669 IC50 = 200 nM T40474 C0DJ2X 44564670 IC50 = 42 nM T40474 CNXH83 44564707 IC50 = 24 nM T40474 C5JQF1 44564752 IC50 = 2000 nM T40474 C4ZM1N 44565117 IC50 = 7.8 nM T40474 C1RO5W 44565118 IC50 = 25 nM T40474 CJD91Q 44565164 IC50 = 28 nM T40474 C2TX8Y 44565165 IC50 = 43 nM T40474 CX06UE 44565221 IC50 = 35 nM T40474 CGM09E 44565222 IC50 = 39 nM T40474 CO75GF 44569268 Ki = 89 nM T40474 CUPE29 44573122 IC50 > 10000 nM T40474 C5JW4L 44573123 IC50 > 10000 nM T40474 C3LI7W 44573124 IC50 = 330 nM T40474 C83MAV 44573125 IC50 > 10000 nM T40474 C1UE4N 44573169 IC50 = 2090 nM T40474 CRB69P 44573170 IC50 = 1950 nM T40474 CHP89M 44573172 IC50 > 10000 nM T40474 CDU37O 44573173 IC50 = 2550 nM T40474 C5EA6B 44573174 IC50 = 340 nM T40474 C0AKT2 44573175 IC50 = 180 nM T40474 CO4P0Q 44573177 IC50 = 130 nM T40474 C23BNM 44573178 IC50 = 5570 nM T40474 CLK94D 44573179 IC50 > 10000 nM T40474 CJAE50 44573180 IC50 > 10000 nM T40474 CL1EB3 44573233 IC50 = 10000 nM T40474 C6WU7Q 44573234 IC50 > 10000 nM T40474 CFR2H7 44573235 IC50 > 10000 nM T40474 CN6ST1 44573237 IC50 = 1590 nM T40474 C54EDN 44573238 IC50 > 10000 nM T40474 CNR7F4 44573242 IC50 > 10000 nM T40474 CE1B0M 44576884 IC50 = 16 nM T40474 CCUR86 44576885 IC50 = 3 nM T40474 C2WE5N 44576886 IC50 = 1 nM T40474 CKJ32O 44576915 IC50 = 4 nM T40474 C3CJ5U 44576916 IC50 = 1 nM T40474 C6Z0QO 44576917 IC50 = 2 nM T40474 CF8I6G 44576918 IC50 = 29 nM T40474 CXD9B4 44578561 IC50 = 850 nM T40474 CA8Y6L 44581208 IC50 = 5000 nM T40474 CV4UO8 44581210 IC50 = 12900 nM T40474 CWVI26 44581243 IC50 = 2000 nM T40474 C0HJ1W 44581292 IC50 = 390 nM T40474 C5D8UH 44581293 IC50 = 170 nM T40474 C2A6VQ 44581294 IC50 = 330 nM T40474 CYV1J0 44581295 IC50 = 1900 nM T40474 CG41XB 44581333 IC50 = 1100 nM T40474 C6HR0S 44581334 IC50 = 7100 nM T40474 C07BKX 44581335 IC50 = 35 nM T40474 C78OMS 44581336 IC50 = 540 nM T40474 CK54XM 44581370 IC50 = 55 nM T40474 CB2H9Z 44581371 IC50 = 320 nM T40474 C9E6LS 44581372 IC50 = 730 nM T40474 CX40GS 44581399 IC50 = 380 nM T40474 CX1O3A 44581670 IC50 = 1300 nM T40474 C6AX3I 44581671 IC50 = 650 nM T40474 CO8N0D 44581673 IC50 = 20100 nM T40474 C87DZS 44581674 IC50 = 5300 nM T40474 CD1QT3 44581709 IC50 = 1300 nM T40474 C3GQN7 44581710 IC50 = 19600 nM T40474 CZMF51 44581711 IC50 = 28300 nM T40474 C1PZ9Q 44581712 IC50 = 3900 nM T40474 CXB64F 44581713 IC50 = 2800 nM T40474 C4CUF5 44581756 IC50 = 5000 nM T40474 COKB58 44581757 IC50 = 60200 nM T40474 CFZ6Y7 44581758 IC50 = 1500 nM T40474 CZ3FU8 44581759 IC50 = 1800 nM T40474 CE30LG 44586566 IC50 = 64 nM T40474 C5K8XT 44586643 IC50 = 7 nM T40474 CZR8A3 44586731 IC50 = 2 nM T40474 C18QMJ 44595039 IC50 = 1.9 nM T40474 C28QLM 44605035 IC50 > 50000 nM T40474 C75XHS 44605037 IC50 > 50000 nM T40474 C32YHG 45102733 IC50 = 3 nM T40474 CU3RF1 45139989 IC50 > 10000 nM T40474 CQGZ06 45139991 IC50 > 10000 nM T40474 C45ZVC 45258276 IC50 = 400 nM T40474 C4K8BX 45267171 IC50 = 26100 nM T40474 C25VIM 45267176 IC50 = 19700 nM T40474 C7RF4H 45267177 IC50 > 40000 nM T40474 CX21TH 45267312 IC50 = 15 nM T40474 C19ODU 45267342 IC50 = 70 nM T40474 CAPB91 45267346 IC50 = 1730 nM T40474 C71UNA 45267350 IC50 = 8100 nM T40474 CH85XT 45267357 IC50 = 20 nM T40474 CTJV09 45267361 IC50 = 16 nM T40474 CV94UD 45268038 IC50 = 12900 nM T40474 CM8Q1I 45268190 IC50 = 5670 nM T40474 C29EHQ 45268213 IC50 = 35 nM T40474 C64DKR 45268916 IC50 = 12500 nM T40474 CLR9Z8 45269054 IC50 = 1700 nM T40474 C4RDV6 45269056 IC50 = 3080 nM T40474 CP17IM 45269085 IC50 = 100 nM T40474 CCQH45 45269092 IC50 = 4400 nM T40474 CDPN59 45269093 IC50 = 25200 nM T40474 C7G9IK 45269098 IC50 = 310 nM T40474 CAC95X 45269918 IC50 = 12100 nM T40474 CE97UZ 45269922 IC50 = 1040 nM T40474 C79COV 45269945 IC50 = 200 nM T40474 CGMC01 45269946 IC50 = 75 nM T40474 CC8X7T 45269953 IC50 = 23 nM T40474 C83VZU 45269959 IC50 = 12 nM T40474 CRC85D 45270590 IC50 = 8600 nM T40474 CIOZ64 45270769 IC50 = 480 nM T40474 CP0TV5 45270775 IC50 = 300 nM T40474 CL90KB 45270780 IC50 = 15 nM T40474 CBI63Q 45270783 IC50 = 11 nM T40474 C9XP0C 45271584 IC50 = 900 nM T40474 CB39AU 45271585 IC50 = 2030 nM T40474 C6PS8T 45271586 IC50 = 20 nM T40474 C36DGY 45272290 IC50 > 40000 nM T40474 COT0W8 45272300 IC50 = 5500 nM T40474 CHN80C 45272463 IC50 = 9 nM T40474 CIQ45M 45272464 IC50 = 15 nM T40474 CZ5MG6 45272468 IC50 = 1880 nM T40474 CMX3S4 45272498 IC50 = 4600 nM T40474 CARY86 45272502 IC50 = 20 nM T40474 CCR6J7 45272508 IC50 = 22 nM T40474 CK7I6J 45272515 IC50 = 14 nM T40474 CC79UA 45273165 IC50 = 12400 nM T40474 CNR8G6 45273175 IC50 > 40000 nM T40474 CHK7B0 45273339 IC50 = 490 nM T40474 C3TQS2 45273344 IC50 = 147 nM T40474 CEI8B2 45381018 Ki = 20 nM T40474 CR6U2Q 45381122 Ki = 13.7 nM T40474 C6E2SC 45482700 IC50 > 10000 nM T40474 CZXH74 45482750 IC50 > 10000 nM T40474 C3VN1M 45483148 IC50 = 7090 nM T40474 CC6X0H 45483156 IC50 = 4270 nM T40474 C2Q0PE 45483158 IC50 = 3330 nM T40474 CRLO64 45483160 IC50 = 3550 nM T40474 C8XMC7 45483167 IC50 = 13680 nM T40474 CYL4E7 45483171 IC50 = 5520 nM T40474 CM15ID 45483173 IC50 = 1210 nM T40474 CT5GL7 45483391 IC50 = 4000 nM T40474 C5FU1M 45483392 IC50 = 30 nM T40474 CM64RU 45483393 IC50 = 40 nM T40474 C24IAB 45483404 IC50 = 200 nM T40474 CN6YG8 45483425 IC50 = 400 nM T40474 CWO2V6 45483426 IC50 = 100 nM T40474 C06MVI 45483427 IC50 = 110 nM T40474 CG50DT 45483428 IC50 = 200 nM T40474 C3R4EO 45483443 IC50 = 60 nM T40474 CK59FA 45483444 IC50 = 30 nM T40474 CDH57Z 45483445 IC50 = 30 nM T40474 CG2XW4 45483457 IC50 = 40 nM T40474 CO5LF4 45483464 IC50 = 50 nM T40474 CF2P7G 45483471 IC50 = 50 nM T40474 C7W6XQ 45483519 IC50 = 40 nM T40474 C8WH4Z 45483526 IC50 = 60 nM T40474 CY9J3H 45483533 IC50 = 50 nM T40474 CGR7H9 45483534 IC50 = 50 nM T40474 CNU1S5 45483535 IC50 = 60 nM T40474 C8KZS7 45487862 IC50 = 7 nM T40474 C98RSQ 45487864 IC50 = 5 nM T40474 CR0X4I 45487870 IC50 = 3 nM T40474 C6C1JY 45488014 IC50 = 23 nM T40474 C4LI7T 45488043 IC50 = 270 nM T40474 C39YHU 45488044 IC50 = 25 nM T40474 C3XTH9 45488051 IC50 = 40 nM T40474 C4MH0A 45488054 IC50 = 870 nM T40474 C53DBE 45488073 IC50 = 65 nM T40474 CL5W8C 45488074 IC50 = 19 nM T40474 CN67YM 45488075 IC50 = 20 nM T40474 C8QIZ1 45488076 IC50 = 36 nM T40474 CZW27U 45488085 IC50 = 36 nM T40474 C0INS5 46194178 IC50 = 48 nM T40474 CUA97D 46209401 IC50 > 10000 nM T40474 CF57GK 46215462 IC50 = 3400 nM T40474 CFS1P2 46218929 IC50 = 7800 nM T40474 CY3HW5 46224684 IC50 > 10000 nM T40474 C2P9QO 46228508 IC50 > 10000 nM T40474 C6E5PY 46228822 IC50 > 10000 nM T40474 C3T8AM 46228951 IC50 > 10000 nM T40474 CYT37A 46232443 IC50 = 130 nM T40474 CG5K2H 46232509 IC50 = 1200 nM T40474 CA98UN 46232510 IC50 = 453 nM T40474 CPK7Z8 46232511 IC50 = 20 nM T40474 C8E4RB 46232512 IC50 = 28 nM T40474 CZ52WR 46232513 IC50 = 59 nM T40474 CAG90T 46232552 IC50 = 205 nM T40474 C1O4DG 46232553 IC50 = 368 nM T40474 CSHX24 46232554 IC50 = 94 nM T40474 C48ZVW 46232555 IC50 = 23 nM T40474 CS9B1U 46232556 IC50 = 9.3 nM T40474 CTYB95 46232607 IC50 = 840 nM T40474 C5KMG3 46232608 IC50 = 2000 nM T40474 CZ90EI 46232636 IC50 > 5000 nM T40474 C7ON5A 46233287 IC50 > 10000 nM T40474 CM58VK 46853747 IC50 = 2 nM T40474 CO8C4F 46853748 IC50 = 3 nM T40474 CYC06D 46862027 IC50 = 2 nM T40474 C9WY1K 46862028 IC50 = 6 nM T40474 CO58RU 46862029 IC50 = 15 nM T40474 CTVI92 46862134 IC50 = 1 nM T40474 C78XDY 46862135 IC50 = 1 nM T40474 COTJ39 46863083 IC50 > 30000 nM T40474 C4EY9T 46864494 IC50 = 1 nM T40474 CE3QM1 46869122 IC50 = 30 nM T40474 CLS29B 46872626 IC50 > 10000 nM T40474 CJOM49 46880136 IC50 = 3100 nM T40474 CRE96X 46885625 IC50 = 316 nM T40474 CT5EO4 46887997 IC50 = 21 nM T40474 CCXK70 46888806 IC50 = 70 nM T40474 C40DPT 46888807 IC50 = 60 nM T40474 CZB8P0 46888808 IC50 = 50 nM T40474 C7K9CZ 46888809 IC50 = 30 nM T40474 C0VSL7 46888810 IC50 = 40 nM T40474 CIXV03 46888811 IC50 = 40 nM T40474 C6UH7Y 46888812 IC50 = 60 nM T40474 C84SJR 46888813 IC50 = 50 nM T40474 CE1JL7 46889250 IC50 = 200 nM T40474 COT4E8 46889251 IC50 > 15000 nM T40474 CQ27HK 46889273 IC50 = 70 nM T40474 C0WYM1 46898022 IC50 = 10000 nM T40474 C97SHZ 46911483 IC50 = 3 nM T40474 CP34VL 46929748 IC50 > 1000 nM T40474 C2B5XF 49765254 IC50 > 10000 nM T40474 CW93FT 49798363 IC50 > 10000 nM T40474 CPBF01 49798365 IC50 = 5200 nM T40474 C9I3KP 49798367 IC50 > 10000 nM T40474 CK8GS3 49798413 IC50 = 1300 nM T40474 CG5YM8 49798415 IC50 = 430 nM T40474 CA2E0R 49798454 IC50 > 10000 nM T40474 CM2T9U 49798477 IC50 = 7 nM T40474 C0DFQ6 49798479 IC50 = 140 nM T40474 CK8H3E 49798481 IC50 = 17 nM T40474 CIE3R8 49798483 IC50 = 60 nM T40474 C2CYA3 49798501 IC50 = 357 nM T40474 C57PFO 49798503 IC50 = 58 nM T40474 C4X0QU 49798505 IC50 = 371 nM T40474 CO3RX7 49798507 IC50 = 26 nM T40474 C0SJ7Q 49804868 IC50 > 5000 nM T40474 CHSF07 49806372 IC50 > 1000 nM T40474 COR4V2 49806718 IC50 > 5000 nM T40474 C5ME3S 49806721 IC50 > 5000 nM T40474 C67HGW 49806722 IC50 > 5000 nM T40474 C8H1FU 49837887 IC50 = 28 nM T40474 CJZ5A0 49840306 IC50 > 10000 nM T40474 CF91RS 49843531 IC50 > 10000 nM T40474 C7EAT8 50898348 IC50 = 42 nM T40474 C2Y6QS 50938552 IC50 > 10000 nM T40474 C82HTZ 50938638 IC50 = 12 nM T40474 CE62UK 50938748 IC50 = 20 nM T40474 CF28WU 50939519 IC50 = 1.87 nM T40474 CTC57I 50940273 IC50 = 23 nM T40474 CX9PS2 50994941 IC50 = 12300 nM T40474 C2V5FL 50996924 IC50 = 166 nM T40474 CM1N2X 50996925 IC50 = 110 nM T40474 C0X9OY 50997095 IC50 = 0.93 nM T40474 CS9G6E 50997096 IC50 = 0.95 nM T40474 COMQ36 50997097 IC50 = 1.01 nM T40474 C8E5QH 50997098 IC50 = 5.6 nM T40474 C96FUK 50997099 IC50 = 230 nM T40474 CIL74P 50997100 IC50 = 10000 nM T40474 CAEI96 50997271 IC50 = 99 nM T40474 CZ9I6X 50997272 IC50 = 2560 nM T40474 CPR8U4 50997273 IC50 = 3440 nM T40474 CSI4X9 50997275 IC50 = 5300 nM T40474 CQTY40 50997276 IC50 = 22400 nM T40474 C83XYM 50997456 IC50 = 12700 nM T40474 C8EY9R 50997457 IC50 = 14300 nM T40474 C6PB0A 50997645 IC50 = 2300 nM T40474 CL0VM3 50997649 IC50 = 1200 nM T40474 CN0D3H 50997650 IC50 = 2.7 nM T40474 CH4G3V 51000498 IC50 = 10 nM T40474 CAZQ43 51003133 IC50 > 1000 nM T40474 C9NYP4 51036677 IC50 > 10000 nM T40474 C4WRY3 51037112 IC50 > 10000 nM T40474 CRI28Z 51037948 IC50 > 10000 nM T40474 C8S4ZV 51038956 IC50 = 7300 nM T40474 C81PZE 51038988 IC50 = 1561 nM T40474 C2GQ8M 51038989 IC50 = 559 nM T40474 CUHG35 51039002 IC50 = 620 nM T40474 CRZ8P7 51039003 IC50 = 760 nM T40474 CH1WR3 52914084 IC50 = 358 nM T40474 C13MUQ 52914647 IC50 = 488 nM T40474 CXA03W 52920796 IC50 > 100 nM T40474 C79CDM 52937011 IC50 = 5800 nM T40474 C45DFE 52937111 IC50 = 10.6 nM T40474 CIW08S 52937112 IC50 = 2.2 nM T40474 C9RHX6 52937192 IC50 = 57 nM T40474 CO37WQ 52937216 IC50 = 450 nM T40474 C8ZH2B 52937217 IC50 = 160 nM T40474 C0H9BK 52937218 IC50 = 3.4 nM T40474 C04PAK 52937219 IC50 = 0.72 nM T40474 CG2M4U 52937323 IC50 = 0.84 nM T40474 C3PLK8 52937324 IC50 = 0.82 nM T40474 C6PM7S 52937325 IC50 = 0.77 nM T40474 CJ89QS 52937326 IC50 = 43 nM T40474 CQT1V8 52937417 IC50 = 4.4 nM T40474 CM24LF 52938983 IC50 = 193.5 nM T40474 C6OTY5 53251320 IC50 > 30000 nM T40474 C09SDH 53257410 IC50 > 10000 nM T40474 CLV61O 53261691 IC50 = 6 nM T40474 CT03OR 53261748 IC50 = 4 nM T40474 CO7MI3 53261751 IC50 = 6 nM T40474 C0YW9C 53261806 IC50 = 26 nM T40474 C9J1LQ 53262468 IC50 = 787 nM T40474 C1H2BK 53262518 IC50 = 5 nM T40474 CUM93B 53262572 IC50 = 227 nM T40474 CJRE96 53262575 IC50 = 11 nM T40474 CXB2N9 53262625 IC50 = 5 nM T40474 CV10UW 53262678 IC50 = 378 nM T40474 C03EDJ 53309832 IC50 > 10000 nM T40474 CTI3K8 53309968 IC50 = 2300 nM T40474 C5MB8L 53309969 IC50 > 10000 nM T40474 C23JMY 53309970 IC50 = 2800 nM T40474 CI0FB1 53309971 IC50 = 770 nM T40474 CATC78 53309972 IC50 = 780 nM T40474 C50GYB 53309973 IC50 > 10000 nM T40474 CAG09D 53309974 IC50 = 1100 nM T40474 C6R9YD 53310117 IC50 = 6100 nM T40474 CE4L6Y 53310118 IC50 = 3000 nM T40474 CPIJ40 53310119 IC50 = 1100 nM T40474 C3W4DE 53310120 IC50 = 440 nM T40474 C0S4WQ 53310121 IC50 = 89 nM T40474 C7MUC4 53310122 IC50 = 790 nM T40474 CZ3I6V 53310262 IC50 = 2000 nM T40474 C2M3PY 53310264 IC50 = 19 nM T40474 CJ68OA 53310395 IC50 = 5 nM T40474 C6QJC9 53310396 IC50 = 11 nM T40474 CQ5V3X 53310397 IC50 = 27 nM T40474 C0J6GA 53310398 IC50 = 9000 nM T40474 C23KML 53310399 IC50 = 9000 nM T40474 C5V0TN 53310400 IC50 = 2300 nM T40474 C41PYS 53310542 IC50 = 31 nM T40474 CYEG47 53310543 IC50 = 2600 nM T40474 CI84VE 53310544 IC50 = 13 nM T40474 CAKF13 53310545 IC50 = 2 nM T40474 CDRI42 53310546 IC50 = 2 nM T40474 C56AOH 53310547 IC50 = 4 nM T40474 C0VSW9 53310688 IC50 = 3 nM T40474 CGV7D0 53310689 IC50 = 3 nM T40474 CO3DU1 53310690 IC50 = 85 nM T40474 C9XSM5 53310691 IC50 = 3 nM T40474 CCK30S 53310692 IC50 = 2 nM T40474 CX10HW 53310824 IC50 = 0.2 nM T40474 C9I0KH 53310825 IC50 = 130 nM T40474 CDT9H2 53310826 IC50 = 3 nM T40474 CLZ60N 53310827 IC50 = 2 nM T40474 C06JVE 53310828 IC50 = 4 nM T40474 CZ6T1A 53310829 IC50 = 75 nM T40474 CE9UD4 53310977 IC50 = 30 nM T40474 C1O8DZ 53310978 IC50 = 10 nM T40474 CCV51N 53310979 IC50 = 5 nM T40474 C38JFV 53310980 IC50 = 3 nM T40474 CR97IC 53310981 IC50 = 2 nM T40474 CI6J2A 53310982 IC50 = 14 nM T40474 C5QFO0 53317399 IC50 = 41 nM T40474 C6E9AG 53317400 IC50 = 32 nM T40474 C8UY3B 53317401 IC50 = 19 nM T40474 CSB19U 53317402 IC50 = 140 nM T40474 C0U6JY 53317525 IC50 = 484 nM T40474 CE8OY2 53317913 IC50 > 100 nM T40474 CGX38E 53318663 IC50 = 56 nM T40474 C2GQS5 53318695 IC50 = 26 nM T40474 CXK28V 53318696 IC50 = 28 nM T40474 CP2ZE6 53318802 IC50 = 10 nM T40474 CR7S3Q 53320012 IC50 = 14 nM T40474 C20IVP 53321284 IC50 = 73 nM T40474 CC63UD 53321285 IC50 = 54 nM T40474 CGPQ42 53321286 IC50 = 203 nM T40474 CMC30H 53321320 IC50 = 50 nM T40474 C09SRW 53321321 IC50 = 30 nM T40474 CNT53F 53321676 IC50 = 47 nM T40474 CYX1F2 53322608 IC50 = 376 nM T40474 CE27TP 53323941 IC50 = 161 nM T40474 C2TCM1 53323942 IC50 = 85 nM T40474 C54YZQ 53323973 IC50 = 17 nM T40474 C2W9OA 53324451 IC50 > 10000 nM T40474 C0XD5M 53325268 IC50 = 24 nM T40474 C9UB7N 53325269 IC50 = 19 nM T40474 CSU20C 53325270 IC50 = 21 nM T40474 C4YG5H 53325271 IC50 = 13 nM T40474 CXOL24 53325517 IC50 = 1652 nM T40474 CO57DC 53325540 IC50 = 45 nM T40474 CI41VZ 53326513 IC50 = 17 nM T40474 CWL68I 53326881 IC50 = 41 nM T40474 C5EOS8 53328013 IC50 = 4100 nM T40474 COJ3C2 53328118 IC50 = 95000 nM T40474 CNET81 53328119 IC50 = 96000 nM T40474 CVC5T4 53328120 IC50 = 36000 nM T40474 C9PR3G 53328121 IC50 = 49000 nM T40474 CG0I5B 53328122 IC50 = 48000 nM T40474 C8WJC1 53328317 IC50 = 14000 nM T40474 C4R1OF 53328318 IC50 > 100000 nM T40474 C2YC0W 53328319 IC50 = 16000 nM T40474 CJIE57 53328320 IC50 = 95000 nM T40474 C6XQ3O 53328321 IC50 > 100000 nM T40474 CKQA18 53328322 IC50 = 13000 nM T40474 CHC90P 53328509 IC50 = 5200 nM T40474 CNG20E 53328510 IC50 = 7600 nM T40474 CA2N6W 53328511 IC50 = 8800 nM T40474 C72RMJ 53328512 IC50 = 27000 nM T40474 C92VPI 53330628 IC50 > 100000 nM T40474 CI23LK 53330629 IC50 > 100000 nM T40474 CEO7M1 53330630 IC50 > 100000 nM T40474 CNPM14 53341082 IC50 > 3000 nM T40474 CM7P3W 53357328 IC50 = 7200 nM T40474 CBK9Q6 53357848 IC50 = 35.7 nM T40474 C4QO8D 53364164 IC50 = 4010 nM T40474 C8NA4L 53384644 IC50 > 30000 nM T40474 C74QJE 53388942 IC50 = 17.38 nM T40474 C35ZPS 53389093 IC50 = 338.84 nM T40474 C60CLS 53389094 IC50 = 562.34 nM T40474 CVG90B 53389651 IC50 > 10000 nM T40474 C8KZ4W 54576161 Ki = 7920 nM T40474 C2FK9I 54576162 Ki = 2820 nM T40474 CIR93L 54576163 Ki = 1710 nM T40474 CV8C3L 54576374 Ki = 6500 nM T40474 CHV91E 54576375 Ki = 2590 nM T40474 CYP5W3 54576376 Ki = 980 nM T40474 C0IU8M 54576377 IC50 = 410 nM T40474 C90PLO 54576378 Ki = 5110 nM T40474 C7B2TQ 54576601 IC50 = 560 nM T40474 C1TX8W 54576602 Ki = 68 nM T40474 CS3D2U 54576603 Ki = 12 nM T40474 CKAP47 54578772 IC50 > 5000 nM T40474 CR9F8Q 54578773 IC50 > 5000 nM T40474 C4Z1NO 54578774 IC50 > 5000 nM T40474 CD6RH1 54578996 IC50 > 5000 nM T40474 CV79SW 54578997 IC50 > 5000 nM T40474 CPZ21F 54579006 Ki = 1980 nM T40474 C9CE8T 54579007 Ki = 240 nM T40474 C9TME2 54579008 IC50 = 740 nM T40474 C89BWQ 54579234 Ki = 201 nM T40474 C58OMU 54579455 Ki = 48.6 nM T40474 C37SZJ 54584802 IC50 > 50000 nM T40474 C8JG9S 54586724 IC50 = 3300 nM T40474 CJ39GM 54757256 IC50 = 330 nM T40474 CE1ZK6 54759168 IC50 > 10000 nM T40474 C9KP8B 54759346 IC50 = 194 nM T40474 CJPV90 54759543 IC50 = 6 nM T40474 CPV0F8 54759721 IC50 = 17 nM T40474 C1XS2J 54760383 IC50 = 6400 nM T40474 CY3V6S 54764326 IC50 = 3 nM T40474 C9ZFS1 54764923 IC50 = 34000 nM T40474 CI79WM 56593141 IC50 = 2.6 nM T40474 CK9JO3 56597774 IC50 = 22 nM T40474 C8AZB0 56597931 IC50 = 28 nM T40474 CM8JX1 56604907 IC50 = 1 nM T40474 C59XFV 56653076 IC50 = 5120 nM T40474 CID82F 56657970 IC50 = 123 nM T40474 C9WA2F 56657971 IC50 = 65.7 nM T40474 CB1DQ4 56657972 IC50 > 10000 nM T40474 CF52XE 56657973 IC50 > 10000 nM T40474 C6DMF7 56658317 IC50 = 6165.95 nM T40474 CJ2I0B 56658318 IC50 = 501.19 nM T40474 CE3A9J 56658438 IC50 = 109.65 nM T40474 C8BSV4 56658439 IC50 = 1071.52 nM T40474 CK4AY2 56658440 IC50 = 3235.94 nM T40474 CQX1B0 56659754 IC50 > 40000 nM T40474 CPEQ43 56659755 IC50 > 40000 nM T40474 CM15EG 56659756 IC50 > 40000 nM T40474 COT59W 56659757 IC50 > 40000 nM T40474 C9JN5I 56659776 IC50 > 40000 nM T40474 CO6XJ2 56659777 IC50 > 40000 nM T40474 CO7N3J 56659778 IC50 > 40000 nM T40474 CR2AZ4 56659779 IC50 > 40000 nM T40474 CR2N6P 56661466 IC50 = 24 nM T40474 CGOX98 56661467 IC50 = 4400 nM T40474 C12SRN 56661502 IC50 = 46.5 nM T40474 CFW6O7 56661504 IC50 > 10000 nM T40474 CL7FE0 56661505 IC50 > 10000 nM T40474 CLI1B7 56661506 IC50 = 69.8 nM T40474 C05DYJ 56661507 IC50 > 10000 nM T40474 CMXJ45 56661685 IC50 = 9600 nM T40474 CWXU56 56661813 IC50 = 108 nM T40474 CN18MD 56661819 IC50 = 13803.84 nM T40474 C6CBL4 56661820 IC50 = 3890.45 nM T40474 CD21PA 56661920 IC50 = 85.11 nM T40474 C5QYO4 56661921 IC50 = 912.01 nM T40474 CLIZ10 56661996 IC50 = 2.5 nM T40474 CIA76R 56662776 IC50 = 130 nM T40474 CP02ZN 56663035 IC50 > 40000 nM T40474 C0TA4N 56663131 IC50 > 40000 nM T40474 C10HLV 56663132 IC50 > 40000 nM T40474 C8CRO9 56663133 IC50 > 40000 nM T40474 CVL35R 56663134 IC50 > 40000 nM T40474 CC6Y5B 56663231 IC50 > 40000 nM T40474 CTPK64 56663250 IC50 > 40000 nM T40474 CWYO21 56663251 IC50 > 40000 nM T40474 CFMW78 56663252 IC50 > 40000 nM T40474 CT7V3Q 56665260 IC50 = 1148.15 nM T40474 C5V7GS 56665261 IC50 = 5495.41 nM T40474 CY5LG6 56665391 IC50 = 54.95 nM T40474 CU24WO 56665392 IC50 = 125.89 nM T40474 CS24OV 56665393 IC50 = 645.65 nM T40474 C8UO0G 56665394 IC50 = 398.11 nM T40474 CUYB95 56665395 IC50 = 9549.93 nM T40474 C0NCP7 56666587 IC50 > 40000 nM T40474 CI9CK1 56666661 IC50 > 40000 nM T40474 CKBD90 56666683 IC50 > 40000 nM T40474 C0Q4XE 56666684 IC50 > 40000 nM T40474 C9J2GI 56668325 IC50 = 300 nM T40474 C2NSX5 56668351 IC50 = 42 nM T40474 CW1F7M 56668352 IC50 = 190.8 nM T40474 CQ0K5X 56668805 IC50 = 1230.27 nM T40474 C3AK9Q 56668822 IC50 = 69.18 nM T40474 CI2J6T 56668823 IC50 = 3548.13 nM T40474 CW4ND5 56668824 IC50 = 2454.71 nM T40474 CM03UF 56668825 IC50 = 1548.82 nM T40474 C9DJH8 56670079 IC50 > 40000 nM T40474 C46PYQ 56670080 IC50 > 40000 nM T40474 C37WLX 56670081 IC50 > 40000 nM T40474 CB83JE 56670082 IC50 > 40000 nM T40474 C8A4RP 56670104 IC50 > 40000 nM T40474 CC54FO 56670105 IC50 > 40000 nM T40474 CJH68T 56671849 IC50 > 10000 nM T40474 CB2HT6 56671943 Ki = 23.7 nM T40474 C0TS2P 56672046 IC50 = 20 nM T40474 C5G0QL 56672191 IC50 = 1621.81 nM T40474 C8SV7G 56672192 IC50 = 2884.03 nM T40474 CN2SU5 56672301 IC50 = 851.14 nM T40474 C4R1GN 56672303 IC50 = 40.74 nM T40474 C8H1RA 56672304 IC50 = 97.72 nM T40474 C9OA3E 56673602 IC50 > 40000 nM T40474 C59WKG 56673603 IC50 > 40000 nM T40474 C4HKA0 56673622 IC50 > 40000 nM T40474 C9TH6I 56673623 IC50 > 40000 nM T40474 CAF70P 56675237 IC50 = 68 nM T40474 CO2V7T 56675238 IC50 > 10000 nM T40474 C3IEZ4 56675239 IC50 > 10000 nM T40474 CI4C3R 56675240 IC50 = 310 nM T40474 C3QA7S 56675566 IC50 = 181 nM T40474 CY4P7C 56675697 IC50 = 154.88 nM T40474 C7MZB1 56675698 IC50 = 125.89 nM T40474 C9ERX0 56675699 IC50 = 426.58 nM T40474 CRJF72 56675700 IC50 = 645.65 nM T40474 CN4O6X 56675701 IC50 = 1348.96 nM T40474 CFC14P 56676919 IC50 > 40000 nM T40474 CXQ3W5 56676939 IC50 > 40000 nM T40474 CS92FR 56676940 IC50 > 40000 nM T40474 C87OYI 56676941 IC50 > 40000 nM T40474 C4ZRM2 56678466 IC50 = 84 nM T40474 CD6FN7 56678556 IC50 > 10000 nM T40474 CA9C0W 56678557 IC50 > 10000 nM T40474 C73ZSK 56678902 IC50 > 100000 nM T40474 CLW26R 56678903 IC50 = 616.6 nM T40474 CQ17GZ 56678904 IC50 = 9549.93 nM T40474 C8GJ3P 56678992 IC50 = 28 nM T40474 C5WUR4 56679001 IC50 = 562.34 nM T40474 C4ARS6 56680232 IC50 > 40000 nM T40474 C7XH1J 56680233 IC50 > 40000 nM T40474 CE8N6R 56680259 IC50 > 40000 nM T40474 CO21ZG 56680260 IC50 > 40000 nM T40474 C86EIX 56680261 IC50 > 40000 nM T40474 C5ZT1C 56681895 IC50 > 10000 nM T40474 CE5QO6 56681896 IC50 > 10000 nM T40474 C7T2EN 56682220 IC50 = 489.78 nM T40474 CI9UG1 56682315 IC50 = 2398.83 nM T40474 CHN09T 56682316 IC50 = 7943.28 nM T40474 CN5W3I 56683485 IC50 > 40000 nM T40474 C8ZJE5 56683588 IC50 > 40000 nM T40474 C5UKI1 56683589 IC50 > 40000 nM T40474 C7Y2EO 56683590 IC50 > 40000 nM T40474 CBOD63 56835089 IC50 > 30000 nM T40474 CR16SD 56947170 IC50 = 1170 nM T40474 CP58NG 56954518 IC50 = 2310 nM T40474 CAK91L 56955954 IC50 > 3600 nM T40474 CWAE98 56970560 IC50 = 793 nM T40474 CPHX64 57325478 IC50 > 50000 nM T40474 CQ9BW4 57325479 IC50 > 50000 nM T40474 CX0D1E 57338725 IC50 = 0.43 nM T40474 CW8A0C 57345939 IC50 = 5920 nM T40474 CM3G0E 57390177 IC50 = 70 nM T40474 C0TM9U 57390203 IC50 = 13 nM T40474 CQF71X 57390565 IC50 = 321 nM T40474 CU0OQ8 57391060 IC50 = 13000 nM T40474 CAE54S 57391542 IC50 = 73 nM T40474 C31NML 57391953 IC50 = 12 nM T40474 CDF6J2 57392000 IC50 = 16 nM T40474 CD2M1W 57393290 IC50 = 27 nM T40474 C0DWE2 57393291 IC50 = 4 nM T40474 COSX75 57393292 IC50 = 3 nM T40474 C2PJN1 57393680 IC50 = 12 nM T40474 CRO72U 57393705 IC50 = 12 nM T40474 C3UHX0 57394704 IC50 > 5000 nM T40474 CH2J1U 57395024 IC50 = 14 nM T40474 CT7MS6 57395025 IC50 = 72 nM T40474 CD6Y9Z 57395116 IC50 > 30000 nM T40474 C8W6IG 57395117 IC50 > 30000 nM T40474 CK1D4R 57395398 IC50 = 34 nM T40474 CV8OD3 57395399 IC50 = 7 nM T40474 CD7C4R 57396463 IC50 > 5000 nM T40474 CTL64V 57396775 IC50 = 29 nM T40474 CFUA48 57396776 IC50 = 5 nM T40474 C4JYZ7 57396777 IC50 = 7 nM T40474 CEQ03L 57396778 IC50 = 5 nM T40474 CG7S0D 57396882 IC50 > 30000 nM T40474 CL8G3R 57397237 IC50 = 17 nM T40474 C24TQU 57398126 IC50 = 15000 nM T40474 C59OYH 57398540 IC50 = 2 nM T40474 CL19DN 57398541 IC50 = 4 nM T40474 CRSL84 57398926 IC50 = 26 nM T40474 CP9W4Y 57399778 IC50 = 4390 nM T40474 CX2UW6 57399904 IC50 > 5000 nM T40474 CE31FR 57399905 IC50 > 5000 nM T40474 CED21U 57400210 IC50 = 3 nM T40474 C35KFY 57400211 IC50 = 3 nM T40474 C0UDY9 57401151 IC50 > 30000 nM T40474 CB02TV 57401549 IC50 = 17000 nM T40474 CJR92U 57401550 IC50 = 1560 nM T40474 C3E4MA 57401677 IC50 > 5000 nM T40474 C51LQS 57402013 IC50 = 27 nM T40474 CZ5VR8 57402451 IC50 = 11 nM T40474 CJF86Y 57402453 IC50 = 18 nM T40474 CI03UC 57403297 IC50 = 227 nM T40474 CP9Z4O 57403409 IC50 > 5000 nM T40474 CRU80Y 57403410 IC50 > 5000 nM T40474 CFXP81 57403758 IC50 = 2 nM T40474 CCT1I4 57403759 IC50 = 4 nM T40474 CR4Y1N 57403760 IC50 = 72 nM T40474 C5K2OW 57405871 IC50 = 0.49 nM T40474 C7YFB3 57405872 IC50 = 6.9 nM T40474 C0BJW4 57405873 IC50 = 2.3 nM T40474 CJ5PK9 57405874 IC50 = 1.2 nM T40474 C9NZK4 57405875 IC50 = 0.46 nM T40474 C1W4CD 57405876 IC50 = 4.1 nM T40474 CZ5XR7 57406042 IC50 = 3.2 nM T40474 C85ICF 57406043 IC50 = 2.3 nM T40474 C7UTX5 57406045 IC50 = 129.2 nM T40474 CVZM52 57406046 IC50 = 126.6 nM T40474 CEP28D 57406047 IC50 = 1.2 nM T40474 C7BX0J 57406219 IC50 = 5.3 nM T40474 CF68ZX 57406220 IC50 = 10.5 nM T40474 C3W6MD 57406221 IC50 = 2 nM T40474 C9WBP0 57406222 IC50 = 2.5 nM T40474 CFHZ69 57406223 IC50 = 4.2 nM T40474 C8D0FL 57406399 IC50 = 2.8 nM T40474 C69LBA 57406400 IC50 = 1.4 nM T40474 CLYG28 57406577 IC50 = 0.19 nM T40474 CS50KZ 57407325 IC50 = 413.2 nM T40474 CZSM95 57412684 IC50 > 10000 nM T40474 CG3EN7 57505462 IC50 = 89 nM T40474 CE59QS 57505507 IC50 > 10000 nM T40474 CV41XZ 57505509 IC50 = 940 nM T40474 C8P6RD 57505528 IC50 > 10000 nM T40474 CHT7S0 57541250 IC50 = 2 nM T40474 CBGY24 57541253 IC50 = 11 nM T40474 C01ANX 57541255 IC50 = 33 nM T40474 C3D8XO 57690955 IC50 = 370 nM T40474 CX1HO9 57691059 IC50 = 9 nM T40474 C74MXU 57691081 IC50 = 31 nM T40474 CBS2Q9 57691146 IC50 = 7 nM T40474 CZ4R8J 57691176 Ki = 4.8 nM T40474 CL6G0X 57691250 IC50 = 7 nM T40474 CORM98 57691278 IC50 = 210 nM T40474 CX3KS5 57691336 Ki = 316 nM T40474 CUCH91 57812280 IC50 = 1600 nM T40474 CR3E0V 57812286 IC50 = 520 nM T40474 CZ0E1D 57812291 IC50 = 2200 nM T40474 CYB5D2 57812313 IC50 = 130 nM T40474 C6JNW5 57812347 IC50 = 42 nM T40474 C2TVB5 57812440 IC50 = 200 nM T40474 CME10V 57812441 IC50 = 190 nM T40474 C3Z5RC 57812480 IC50 = 30 nM T40474 C90UAY 57812481 IC50 = 2100 nM T40474 CF94GH 57812483 IC50 = 86 nM T40474 CSWG27 57812520 IC50 = 290 nM T40474 CK1M2H 57812531 IC50 = 430 nM T40474 C6DS4B 57812548 IC50 = 7400 nM T40474 C13ZEB 57812551 IC50 = 550 nM T40474 CWYI07 57812563 IC50 = 950 nM T40474 C29DUL 57812564 IC50 = 220 nM T40474 CJ1Q9W 57812570 IC50 = 110 nM T40474 CK2ZA8 57812588 IC50 = 130 nM T40474 C4ED9U 57812594 IC50 = 590 nM T40474 C2BR4G 57812601 IC50 = 560 nM T40474 CT7UW0 57812618 IC50 = 260 nM T40474 CZ0Y3X 57812627 IC50 = 360 nM T40474 C1NC3Y 57812678 IC50 = 780 nM T40474 CJM13Z 57812755 IC50 = 320 nM T40474 CQ6XH9 57812769 IC50 = 590 nM T40474 C3HS4R 58015489 IC50 = 2 nM T40474 CVK0G4 58056356 IC50 > 50000 nM T40474 C3VI7D 58229394 IC50 = 338 nM T40474 CNXU29 58229412 IC50 = 1307 nM T40474 C52OMW 58229434 IC50 = 609 nM T40474 C7HPC2 58268648 Ki = 2.3 nM T40474 CC79OM 58270290 IC50 = 5 nM T40474 CR7L0J 58955249 IC50 = 44 nM T40474 C6BPR2 58985201 IC50 > 30000 nM T40474 CL82WA 59320262 Ki = 89.7 nM T40474 CWX3N7 59320301 Ki = 4 nM T40474 C82LMW 59341790 IC50 = 35.6 nM T40474 C60WQR 59341800 Ki = 20.9 nM T40474 CTC3Q7 59341811 Ki = 15 nM T40474 C1CM7K 59341825 Ki = 6 nM T40474 C39PBN 59341841 Ki = 44 nM T40474 COE1A5 59341845 IC50 = 17 nM T40474 C0EP5I 59341847 IC50 = 0.7 nM T40474 C74MWB 59341863 Ki = 34 nM T40474 CCRG83 59341868 IC50 = 16 nM T40474 C0EYG8 59341873 Ki = 140 nM T40474 CRHS79 59341881 Ki = 4 nM T40474 CUQ5X1 59341900 Ki = 9 nM T40474 CO6CT8 59341929 Ki = 61.7 nM T40474 CR8UM2 59341930 Ki = 106 nM T40474 C6HG2C 59341933 Ki = 68 nM T40474 C87RPJ 59341936 Ki = 4.8 nM T40474 C4MHN9 59341953 IC50 = 25 nM T40474 CHQ28A 59341978 IC50 = 0.5 nM T40474 CRF09L 59484839 IC50 = 2.7 nM T40474 C7B5MJ 59484894 IC50 = 200 nM T40474 CR3UX7 59484959 IC50 < 1 nM T40474 CJ03ZP 59534523 IC50 = 2100 nM T40474 CX9B7L 59534559 IC50 > 30000 nM T40474 C1CLT5 59534567 IC50 = 400 nM T40474 C1E3OI 59598370 Ki = 1.1 nM T40474 CQ2UE7 59598391 Ki = 1.3 nM T40474 C5AEN1 59598393 Ki = 16.7 nM T40474 CUA1F5 59598396 Ki = 1.9 nM T40474 C0O6ZX 59598404 Ki = 0.9 nM T40474 CBMH78 59598415 Ki = 1.4 nM T40474 CYNP39 59598421 Ki = 1.4 nM T40474 CU1ER8 59598432 Ki = 0.8 nM T40474 C0L5DN 59598437 Ki = 0.9 nM T40474 CKVB01 59598456 Ki = 0.6 nM T40474 CXJ63M 59603829 IC50 = 4000 nM T40474 CQEU96 59603842 IC50 = 410 nM T40474 CDW76U 59849751 IC50 = 90 nM T40474 CL9UP8 59849760 IC50 = 11 nM T40474 CCX2Q5 59864465 Ki = 1.2 nM T40474 CYTO24 60142557 IC50 = 28 nM T40474 C23JEF 60142558 IC50 = 210 nM T40474 C6DHB7 60142693 IC50 = 130 nM T40474 C1FOD2 60142694 IC50 = 45 nM T40474 C54MUW 60142695 IC50 = 88 nM T40474 CP3NW0 60142697 IC50 = 67 nM T40474 C7V6CZ 60142827 IC50 = 41 nM T40474 C3JE8D 60142953 IC50 = 27 nM T40474 CBCE37 60142954 IC50 = 180 nM T40474 C6XA7U 60142955 IC50 = 9 nM T40474 C36JUG 60143085 IC50 = 3 nM T40474 CL0N9F 60143086 IC50 = 0.2 nM T40474 CZT65A 60143089 IC50 = 48 nM T40474 CSZA16 60155724 IC50 > 3600 nM T40474 CK8EN9 60166357 IC50 = 92 nM T40474 CX7U4D 60168372 IC50 = 20 nM T40474 C9ZCT2 62705065 IC50 = 7.7 nM T40474 C6RNA3 66548952 IC50 = 101.7 nM T40474 CJ9Y6E 66548953 IC50 = 171.4 nM T40474 CJ04HQ 66548954 IC50 = 16.4 nM T40474 C3VZI6 66549137 IC50 = 61.8 nM T40474 C5C8EH 66549322 IC50 = 44.9 nM T40474 C1NOI9 66549323 IC50 = 45.3 nM T40474 C5JUW4 66549324 IC50 = 22.1 nM T40474 CW4CN2 66549325 IC50 = 101 nM T40474 CVCT83 66549326 IC50 = 25.8 nM T40474 C3OT0Y 66549510 IC50 = 44.9 nM T40474 CLB71O 66549513 IC50 = 76.8 nM T40474 CGF64K 66549695 IC50 = 81.7 nM T40474 C5YMQ0 66549698 IC50 = 26.5 nM T40474 CWR3E4 66549699 IC50 = 151.8 nM T40474 COX03B 66549892 IC50 = 50.5 nM T40474 CHNX35 66549893 IC50 = 66.2 nM T40474 CWJ1Q8 66549894 IC50 = 130.2 nM T40474 CD2M3B 66549895 IC50 = 21.4 nM T40474 CN9VC1 66549896 IC50 = 228.7 nM T40474 CUK53J 66550108 IC50 = 58.7 nM T40474 CKV6O2 66550109 IC50 = 228.3 nM T40474 CCM2D3 66550111 IC50 = 320 nM T40474 CZ5I4W 66550112 IC50 = 99 nM T40474 C4GX0I 66550113 IC50 = 510 nM T40474 C3G7YV 66550333 IC50 = 210 nM T40474 CZ5G7S 66550334 IC50 = 340 nM T40474 C8UFL9 66550335 IC50 = 1140 nM T40474 CX41BC 66550336 IC50 = 19.4 nM T40474 CDY29W 66553435 IC50 = 1200 nM T40474 C5B9TI 66553436 IC50 = 7000 nM T40474 CCO23J 66553437 IC50 = 600 nM T40474 C69XTG 66553438 IC50 = 4110 nM T40474 C5LVX0 66553439 IC50 = 480 nM T40474 CKT0N7 66553440 IC50 = 1300 nM T40474 CUD21N 66553441 IC50 = 1140 nM T40474 C3XM5A 66553506 IC50 = 410 nM T40474 C1GUI3 66553507 IC50 = 560 nM T40474 C7XA1P 66553511 IC50 = 280 nM T40474 C10AMI 66553589 IC50 = 22 nM T40474 CN9SC4 66968949 IC50 = 1.7 nM T40474 C1HSE0 67035086 IC50 > 10000 nM T40474 CWI6K5 67035106 IC50 > 10000 nM T40474 C38RGB 67035556 IC50 > 10000 nM T40474 CD14OC 67071561 IC50 = 1535 nM T40474 CEKN37 67073846 IC50 = 127 nM T40474 C37NKO 67129970 IC50 > 10000 nM T40474 CK80LJ 67130050 IC50 > 10000 nM T40474 CV63UL 67240318 IC50 > 10000 nM T40474 C19FHU 67388618 IC50 = 240 nM T40474 CMLP73 67404214 IC50 = 89 nM T40474 C8COE7 67455704 Ki = 6.14 nM T40474 C6TO0M 68287716 IC50 = 359 nM T40474 CT35XG 68288060 IC50 = 130 nM T40474 C75XZR 68288074 IC50 = 142 nM T40474 CY5I9P 68289004 IC50 = 12 nM T40474 CK7ZE3 68289353 IC50 = 24 nM T40474 CF5Q9D 68289397 IC50 = 27 nM T40474 C8I7GC 68293638 IC50 > 10000 nM T40474 CD56XK 68293660 IC50 > 10000 nM T40474 C87LEP 68353938 IC50 = 9 nM T40474 C3U8AY 68353940 IC50 = 6 nM T40474 CI9NA6 68353946 IC50 = 13 nM T40474 C7CVF6 68353953 IC50 = 20 nM T40474 CNF02U 68353989 IC50 = 32 nM T40474 C9YDO2 68353991 IC50 = 3 nM T40474 C81QAH 68355550 IC50 = 6 nM T40474 CCL3H8 68505435 IC50 = 4200 nM T40474 C61KMD 68506553 IC50 = 6.5 nM T40474 C6VIK8 68508446 IC50 = 10 nM T40474 C9M3JV 68509959 IC50 = 1 nM T40474 CQ2OL5 68512172 IC50 > 1 nM T40474 C7GRV2 68755406 IC50 > 10000 nM T40474 C5DGR9 69036886 IC50 = 1247 nM T40474 C0F3ZG 70677252 Ki = 19.8 nM T40474 CK6GF8 70677253 Ki = 69 nM T40474 CPSZ68 70677254 Ki = 379 nM T40474 CD02XA 70677255 Ki = 51.8 nM T40474 C23VPA 70677256 Ki = 6510 nM T40474 C71EUH 70677257 Ki = 7390 nM T40474 C3NKD1 70677258 Ki = 425 nM T40474 CN3U5G 70677395 Ki = 188 nM T40474 CR50BQ 70677396 Ki = 2 nM T40474 C1MSX9 70677397 IC50 = 5 nM T40474 C06LOZ 70677398 Ki = 4 nM T40474 CA2C6M 70677399 Ki = 73 nM T40474 CL3KD5 70677400 Ki = 653 nM T40474 CE8A6S 70677533 IC50 = 51 nM T40474 CWS08A 70677534 Ki = 35 nM T40474 CNHC64 70678116 IC50 > 50000 nM T40474 CUEO45 70681644 Ki = 5.1 nM T40474 CY7DW8 70681656 IC50 = 34 nM T40474 C1YH4R 70681671 IC50 = 28 nM T40474 CL3AG5 70681673 IC50 = 14 nM T40474 C59QUO 70683775 Ki = 12.8 nM T40474 C3RQ0D 70683776 Ki = 28.4 nM T40474 CTO9G0 70683779 Ki = 56.7 nM T40474 CZ8L2W 70683780 Ki = 60.2 nM T40474 C0J7UE 70683787 IC50 = 77 nM T40474 CE8WY0 70685920 Ki = 140 nM T40474 C3O4UL 70688040 Ki = 22 nM T40474 C4BLJ8 70688051 IC50 = 1.6 nM T40474 CSB69C 70688053 IC50 = 130 nM T40474 C3NHX5 70688055 IC50 = 150 nM T40474 CU02FW 70688063 IC50 = 51 nM T40474 CNYI07 70688065 IC50 = 53 nM T40474 C4CY2F 70690067 Ki = 3.4 nM T40474 CL0F7V 70690072 Ki = 1.6 nM T40474 C7I6QX 70690073 Ki = 4.4 nM T40474 CN8F4V 70690082 IC50 = 23 nM T40474 C3OVZ0 70692216 Ki = 1.9 nM T40474 CLZ65T 70692217 Ki = 7.2 nM T40474 CQIB46 70692219 Ki = 37.8 nM T40474 CO5JY8 70692223 IC50 = 63 nM T40474 CHAC25 70694313 IC50 = 90 nM T40474 C97MNY 70694315 IC50 = 220 nM T40474 CCE3X9 70696383 IC50 = 800 nM T40474 CU3NZ7 70696384 IC50 = 130 nM T40474 CH0KU1 70696392 IC50 = 110 nM T40474 CF9H7K 70696395 IC50 = 4 nM T40474 C8T7ZP 70789255 IC50 = 183000 nM T40474 CH0B8N 70789756 IC50 = 4510 nM T40474 C9GUM2 70811848 IC50 = 240.3 nM T40474 C23VCD 70988670 IC50 = 1.7 nM T40474 C6BJ8T 71148152 Ki = 250 nM T40474 CTE9X7 71148153 Ki = 379 nM T40474 CN0EA5 71449347 IC50 = 659 nM T40474 CS51JQ 71449348 IC50 = 879 nM T40474 CJ1OK7 71449349 IC50 = 6.5 nM T40474 C6D4VB 71451155 IC50 = 2500 nM T40474 CYR2A7 71451157 IC50 = 485 nM T40474 CEBO91 71452977 IC50 = 3900 nM T40474 CE09IP 71452979 IC50 = 309 nM T40474 CV75CT 71452980 IC50 = 539 nM T40474 CUJO06 71452981 IC50 > 10 nM T40474 C2SU6A 71454728 IC50 = 2700 nM T40474 C05MOI 71454729 IC50 = 1980 nM T40474 C31BZW 71454730 IC50 > 10 nM T40474 C2SRG8 71454731 IC50 = 441 nM T40474 CKT60L 71455860 Ki = 1600 nM T40474 CS5O0Z 71456479 IC50 = 441 nM T40474 C48DBN 71456480 IC50 = 385 nM T40474 CTX26B 71456481 IC50 = 924 nM T40474 CVA93Y 71458337 IC50 = 486 nM T40474 CKU6H3 71460177 IC50 = 626 nM T40474 CX4PH7 71461890 IC50 = 409 nM T40474 C65GYB 71461891 IC50 = 257 nM T40474 C6Q2RP 71461892 IC50 > 10 nM T40474 CGNJ74 71461893 IC50 > 1000 nM T40474 C6E7JR 71492737 IC50 = 850 nM T40474 C5X2GS 71493611 IC50 = 390 nM T40474 CULK13 71493612 IC50 = 460 nM T40474 CV0ZG4 71493613 IC50 = 280 nM T40474 CSEA28 71493749 IC50 = 430 nM T40474 C6BZ3F 71493750 IC50 = 1230 nM T40474 C27BMG 71493896 IC50 = 570 nM T40474 C9SB8Y 71493897 IC50 = 210 nM T40474 CD0B9W 71493898 IC50 = 240 nM T40474 CAW17X 71494057 IC50 = 45 nM T40474 CQKT80 71494059 IC50 = 550 nM T40474 C1WK8N 71494060 IC50 = 280 nM T40474 CLCK46 71494223 IC50 = 340 nM T40474 CDE4X6 71494225 IC50 = 5 nM T40474 C10RDA 71494226 IC50 = 150 nM T40474 CRQH48 71494227 IC50 = 99 nM T40474 C6X8JW 71494394 IC50 = 210 nM T40474 CC67KE 71494395 IC50 = 120 nM T40474 CVK6Y7 71494534 IC50 > 25000 nM T40474 C92DXO 71494535 IC50 > 25000 nM T40474 C0Y7IK 71494536 IC50 > 25000 nM T40474 CF8G2R 71494537 IC50 > 25000 nM T40474 CIA18Y 71494686 IC50 > 25000 nM T40474 CG4HP9 71497990 IC50 = 5.92 nM T40474 C1KB2U 71497991 IC50 = 6.68 nM T40474 C92XST 71498012 IC50 = 4.8 nM T40474 CR0QM2 71498048 IC50 = 27.49 nM T40474 CQY31T 71498139 IC50 = 0.59 nM T40474 CJF70K 71498153 IC50 = 1.65 nM T40474 CD4T2R 71498154 IC50 = 2.76 nM T40474 C0LY6D 71498155 IC50 = 1.03 nM T40474 C8IU2T 71498156 IC50 = 1.22 nM T40474 CV7CH3 71498171 IC50 = 3.13 nM T40474 C5VQ3T 71498174 IC50 = 3.02 nM T40474 C5ZA7L 71498190 IC50 = 2.72 nM T40474 CZ16VL 71498192 IC50 = 3.55 nM T40474 C0ID5P 71498193 IC50 = 1.05 nM T40474 CE3I0U 71498211 IC50 = 2.64 nM T40474 CWH20D 71498234 IC50 = 13.5 nM T40474 C0G9JD 71498258 IC50 = 4.5 nM T40474 CP6C4I 71498279 IC50 = 8.42 nM T40474 C64ZAV 71498281 IC50 = 5.23 nM T40474 CB8ZX2 71510447 IC50 = 1.5 nM T40474 C1V0AY 71510450 IC50 = 151.9 nM T40474 CB1CQ7 71510572 IC50 = 664.2 nM T40474 CT04AM 71510706 IC50 = 418.8 nM T40474 C1KC5A 71510707 IC50 = 116.7 nM T40474 CAO04I 71510709 IC50 = 103 nM T40474 C4G2UN 71510710 IC50 = 192 nM T40474 CG9VD1 71510856 IC50 = 132.5 nM T40474 CZ4M5S 71511128 IC50 = 2.4 nM T40474 C9DIK2 71512060 IC50 > 10000 nM T40474 CY4OQ9 71515572 IC50 = 1500 nM T40474 C9V5YC 71515573 IC50 = 1600 nM T40474 CG4HU8 71515638 IC50 = 100 nM T40474 CVU65I 71515639 IC50 = 900 nM T40474 CSE95N 71515705 IC50 = 200 nM T40474 CT1Q8V 71515973 IC50 = 583 nM T40474 CK9R7M 71515974 IC50 = 85 nM T40474 CEC25B 71516026 IC50 = 151 nM T40474 C5D1WP 71516156 IC50 > 10000 nM T40474 C0LZN7 71516421 IC50 = 360 nM T40474 C56QVR 71516422 IC50 = 1000 nM T40474 CAQM32 71516423 IC50 = 210 nM T40474 CW7O9R 71516496 IC50 = 160 nM T40474 C4N9IP 71516499 IC50 = 300 nM T40474 CP9VK4 71528197 IC50 = 2600 nM T40474 CCN01X 71547862 IC50 > 10000 nM T40474 CA3O6K 71552696 IC50 = 10320 nM T40474 C1NPL0 71552941 IC50 = 5070 nM T40474 CA4PS8 71552942 IC50 = 6000 nM T40474 CL3VD5 71579695 IC50 = 8000 nM T40474 C1BCX0 71579696 IC50 = 12 nM T40474 CA3BJ7 71579697 IC50 = 31 nM T40474 C85QGV 71579785 IC50 = 78 nM T40474 CG27VX 71579787 IC50 = 24 nM T40474 CIKO04 71579788 IC50 = 152 nM T40474 C9FKI7 71579789 IC50 = 76 nM T40474 CYMB89 71579879 IC50 = 48 nM T40474 CDI95L 71579880 IC50 = 142 nM T40474 CL87FP 71579881 IC50 = 23 nM T40474 C39NKW 71579882 IC50 = 75 nM T40474 CM8F7R 71579883 IC50 = 27 nM T40474 CDZ9U3 71579967 IC50 = 30 nM T40474 CZO62R 71579968 IC50 = 27 nM T40474 CW19HG 71579969 IC50 = 14 nM T40474 C2HOR9 71579970 IC50 = 0.32 nM T40474 CZ31PU 71583657 IC50 = 5600 nM T40474 C5QTH7 71601341 IC50 = 190 nM T40474 C3X6YG 71601483 IC50 = 1 nM T40474 CED8U9 71601485 IC50 = 60 nM T40474 C9JZ5E 71601486 IC50 = 1888 nM T40474 CXLQ94 71601487 IC50 = 1157 nM T40474 CG1MR6 71601488 IC50 = 3691 nM T40474 CHA9O3 71601634 IC50 = 94 nM T40474 CB8JI6 71601635 IC50 = 3191 nM T40474 C8O2PF 71601636 IC50 = 1368 nM T40474 CBSF14 71601639 IC50 = 70 nM T40474 C0VOJ8 71601790 IC50 = 32 nM T40474 CN2W0E 71601934 IC50 = 53 nM T40474 C6FH5O 71601935 IC50 = 14 nM T40474 C1LT7J 71602068 IC50 = 5 nM T40474 CJ1VR4 71602069 IC50 = 3 nM T40474 C7LOM2 71602070 IC50 = 67 nM T40474 C9ULZ6 71602071 IC50 = 55 nM T40474 CXNG24 71622198 IC50 = 9.8 nM T40474 CX7F5R 71625135 IC50 = 9500 nM T40474 C9UZN6 71625137 IC50 = 8400 nM T40474 CGD80H 71625269 IC50 = 4300 nM T40474 C8KWL0 71625388 IC50 = 1200 nM T40474 CTX12L 71625497 IC50 = 6600 nM T40474 CGR0S1 71625499 IC50 = 4000 nM T40474 CQ5XN2 71625729 IC50 = 4300 nM T40474 C02ZVM 71658195 IC50 = 14.5 nM T40474 C08RAB 71658196 IC50 = 5.08 nM T40474 C1AWG8 71658328 IC50 = 5.05 nM T40474 C0WUN9 71658329 IC50 = 3.4 nM T40474 C1P8ZY 71658330 IC50 = 18.4 nM T40474 C1LQ5N 71658331 IC50 = 4.12 nM T40474 CMPE61 71658471 IC50 = 11.9 nM T40474 CMBV96 71658472 IC50 = 10.4 nM T40474 C0S5DX 71658473 IC50 = 3.64 nM T40474 C7IQ2H 71658474 IC50 = 10.24 nM T40474 CHE4B8 71658607 IC50 = 24.35 nM T40474 CR1S9H 71658608 IC50 = 21.12 nM T40474 CW25GT 71658609 IC50 = 20.57 nM T40474 C2YEV0 71666369 IC50 = 7.8 nM T40474 CIK9T6 71666371 IC50 = 1.8 nM T40474 CH9Y3P 71666520 IC50 = 2.7 nM T40474 CS42GU 71666523 IC50 = 2180 nM T40474 CD3BA9 71666670 IC50 = 6 nM T40474 C06LAC 71666672 IC50 = 2 nM T40474 CX6BR2 71666816 IC50 = 2.4 nM T40474 C6B4SW 71666818 IC50 = 39.1 nM T40474 CCF57W 71666819 IC50 = 4.2 nM T40474 C36ACQ 71666955 IC50 = 21.4 nM T40474 C9X8SD 71666958 IC50 = 3.4 nM T40474 CZF3M6 71667102 IC50 = 0.7 nM T40474 CV9X4J 71667249 IC50 = 0.9 nM T40474 CD9Z3P 71667252 IC50 = 11.1 nM T40474 CZO59L 71677856 IC50 = 16.83 nM T40474 CP9C1O 71678016 IC50 = 270 nM T40474 C1KL8U 71678017 IC50 = 380 nM T40474 CG39HK 71678357 IC50 = 280 nM T40474 C2XGC7 71678520 IC50 = 230 nM T40474 CO2G7N 71678692 IC50 = 210 nM T40474 CIH6U9 71678693 IC50 = 920 nM T40474 C3T1HM 71678864 IC50 > 10000 nM T40474 C1Z7OI 71678868 IC50 = 32 nM T40474 C7AG6Y 71679031 IC50 = 21 nM T40474 CCL68Y 71679032 IC50 = 56 nM T40474 C48WGO 71679034 IC50 = 29 nM T40474 CY2T4W 71679036 IC50 = 46 nM T40474 CXC91N 71679037 IC50 = 38 nM T40474 C3N5CO 71679200 IC50 = 49 nM T40474 CO6DZ4 71679365 IC50 = 19 nM T40474 CJL7U4 71679366 IC50 = 18 nM T40474 CGHY50 71679368 IC50 = 26.26 nM T40474 C1FAU8 71679855 IC50 = 1.4 nM T40474 C1N3QC 71680199 IC50 = 4.4 nM T40474 CI09HT 71680564 IC50 = 13700 nM T40474 CC1O7E 71697465 IC50 = 2.64 nM T40474 CZ0MR2 71697565 IC50 = 1.32 nM T40474 CUI1D3 71697780 IC50 = 3.13 nM T40474 CW39CL 71697781 IC50 = 2.72 nM T40474 CVZW80 71697883 IC50 = 3.45 nM T40474 CZ63CK 71698087 IC50 = 1.65 nM T40474 C2AR4U 71717471 IC50 = 10 nM T40474 C45LSX 71720501 IC50 = 8 nM T40474 CJY74A 71727182 IC50 = 330 nM T40474 C9KA2V 71739682 IC50 = 420 nM T40474 CN53MG 71739683 IC50 = 290 nM T40474 CHS3G4 71739810 IC50 = 380 nM T40474 C2O6YP 71739811 IC50 = 170 nM T40474 C6M2SA 71739812 IC50 = 640 nM T40474 C8XL6J 71739813 IC50 = 37000 nM T40474 CD1C0F 71739814 IC50 = 450 nM T40474 CE1CU3 71739815 IC50 = 830 nM T40474 C8P1QI 71739937 IC50 = 19000 nM T40474 CQP31V 71739938 IC50 = 580 nM T40474 CN5PK2 71769802 IC50 = 26 nM T40474 CV6G2Q 71769803 IC50 = 13 nM T40474 CP17NV 71769804 IC50 = 4.4 nM T40474 CTJA64 71769805 IC50 = 3.9 nM T40474 CQBY96 71769920 IC50 = 43 nM T40474 C6E9RL 71769921 IC50 = 24 nM T40474 C18SQD 71769922 IC50 = 22 nM T40474 C7Y5NZ 71769923 IC50 = 35 nM T40474 CT5W6X 71770050 IC50 = 12 nM T40474 C8EY0X 71770052 IC50 = 190 nM T40474 C6MF1E 71770053 IC50 = 61 nM T40474 C4PBI1 71770186 IC50 = 91 nM T40474 CDC0E7 71770188 IC50 = 940 nM T40474 C01BGH 71770189 IC50 = 120 nM T40474 CO5YA4 71770190 IC50 = 43 nM T40474 CU8HP7 71770314 IC50 = 110 nM T40474 C8HLV2 71770315 IC50 = 95 nM T40474 CLM10P 71770316 IC50 = 22 nM T40474 CD1TG8 71770432 IC50 = 26 nM T40474 CZ3GD0 71770433 IC50 = 34 nM T40474 CTM38H 71770435 IC50 = 5.3 nM T40474 CB0Z7L 71770555 IC50 = 120 nM T40474 CA0P8K 72164291 IC50 > 10000 nM T40474 C26SBP 72164410 IC50 = 9000 nM T40474 CTJH89 72190201 IC50 = 5 nM T40474 C8Z1RG 72190203 IC50 = 2 nM T40474 CI73EM 72190518 IC50 = 12 nM T40474 C7B1HQ 72190519 IC50 = 35 nM T40474 C5W9RJ 72190521 IC50 = 10 nM T40474 CXP6Q0 72190522 IC50 = 55 nM T40474 CJN19P 72190820 IC50 = 11 nM T40474 C6V8HW 72190821 IC50 = 21 nM T40474 C0QS1P 72190823 IC50 = 27 nM T40474 CCUO41 72191120 IC50 = 16 nM T40474 CP2YF5 72191121 IC50 = 7 nM T40474 C6XFD2 72191122 IC50 = 9 nM T40474 CZY7H6 72191430 IC50 = 21 nM T40474 CVJ5T7 72191431 IC50 = 19 nM T40474 C5VWC1 72191432 IC50 = 7 nM T40474 CSRB27 72191744 IC50 = 3 nM T40474 C2O3EA 72192349 IC50 = 28 nM T40474 C46UJE 72192350 IC50 = 90 nM T40474 C8L3AD 72192351 IC50 = 8 nM T40474 C3Y8WU 72192352 IC50 = 40 nM T40474 CJ7QW9 72192645 IC50 = 5 nM T40474 CD50ES 72204020 IC50 = 38.1 nM T40474 C6Q5OT 72204188 IC50 = 64.9 nM T40474 C7OQ1U 72204189 IC50 = 97.9 nM T40474 CD7Q3B 72204190 IC50 = 196.4 nM T40474 C6RLG8 72204191 IC50 = 173.2 nM T40474 C9J4UC 72699437 IC50 = 49.7 nM T40474 C1DMB4 72737557 IC50 = 330 nM T40474 CH8I6T 72737558 IC50 = 2.3 nM T40474 C52VCP 72737559 IC50 = 5.2 nM T40474 CIZC74 73211773 IC50 > 1000 nM T40474 CBM61I 73293715 Ki = 4 nM T40474 CC6NH1 73293716 Ki = 4 nM T40474 CF90CM 73293717 Ki = 3 nM T40474 CIV18Y 73293899 Ki = 5 nM T40474 CU74EN 73293900 IC50 = 5 nM T40474 CQ5U3W 73293901 Ki = 4 nM T40474 CJ0IW9 73293902 Ki = 7 nM T40474 C6NB5X 73293903 Ki = 24 nM T40474 CHMY19 73293904 Ki = 12 nM T40474 C17TVK 73294098 Ki = 8 nM T40474 C1HG4W 73294099 Ki = 10.1 nM T40474 CA2J1Q 73294100 Ki = 16.7 nM T40474 CT49KB 73347899 IC50 = 7.96 nM T40474 CD2XO5 73347902 IC50 = 6.23 nM T40474 CKUR19 73348870 IC50 = 7.54 nM T40474 C0RP6H 73349432 IC50 = 9.37 nM T40474 C8SIL6 73349435 IC50 = 1.39 nM T40474 C56VXD 73352475 IC50 = 4.48 nM T40474 C1ILQ2 73355484 IC50 = 16.36 nM T40474 CV8L5P 73355489 IC50 = 12.64 nM T40474 CF9C0A 73386808 IC50 > 1000 nM T40474 CVNW01 73386831 IC50 = 0.84 nM T40474 C9HNZ4 73387103 IC50 > 1000 nM T40474 C96XKM 73387105 IC50 > 1000 nM T40474 CQ48ZS 73387126 IC50 = 4.6 nM T40474 C1V3NZ 73425588 IC50 = 364 nM T40474 C3UC9H 73891099 IC50 = 580 nM T40474 C3E9MB 76281906 IC50 = 6 nM T40474 CAZ5N3 76281907 IC50 = 63 nM T40474 CTKJ62 76281908 IC50 = 13 nM T40474 C19PGZ 76282166 IC50 = 2.4 nM T40474 CTEF85 76282167 IC50 = 6.4 nM T40474 CC2K0H 76282402 IC50 > 1000 nM T40474 CEW67B 76282644 IC50 = 7.2 nM T40474 CV8QX0 76310169 IC50 = 9650 nM T40474 CA5L4W 76324771 IC50 > 30000 nM T40474 C9GO0P 76328313 IC50 = 8630 nM T40474 C4K6IE 76335350 IC50 = 39 nM T40474 C39FTZ 76335685 IC50 > 100000 nM T40474 CH8W7D 77461036 IC50 = 153 nM T40474 CHLR89 78673838 IC50 = 6.7 nM T40474 C0QK9F 86288869 IC50 = 398 nM T40474 C06BFO 86288903 IC50 = 0.9 nM T40474 CZ73DG 86288904 IC50 = 1.7 nM T40474 C83GTK 86291722 IC50 = 122.7 nM T40474 CN84BH 86291723 IC50 = 37 nM T40474 C7PE9O 86291932 IC50 = 42.5 nM T40474 C9PQ8Y 86291933 IC50 = 12 nM T40474 C2VF0H 86292125 IC50 = 9.3 nM T40474 CNB6W9 86292126 IC50 = 7.9 nM T40474 CO1Z8Y 86292127 IC50 = 20.1 nM T40474 CBY03E 86292128 IC50 = 11.4 nM T40474 CPG3A5 86302574 IC50 = 0.7 nM T40474 C6LQR8 86566404 EC50 = 190.3 nM T40474 CK5M2N 86566405 EC50 = 155.4 nM T40474 C79QGH 86566406 EC50 = 278.7 nM T40474 COA60C 86566407 EC50 = 133.8 nM T40474 CI84CJ 86566427 EC50 > 1000 nM T40474 CN6WR8 86566539 EC50 = 1.8 nM T40474 C09AGQ 86566540 EC50 = 1.6 nM T40474 CVP92Y 86566542 EC50 = 1.3 nM T40474 C3RVG2 86566598 EC50 = 23.8 nM T40474 CK79PB 86566601 EC50 = 4.9 nM T40474 CZ9S6H 86566631 EC50 = 38.1 nM T40474 CC48MV 86566650 EC50 = 9.9 nM T40474 CO47CE 86566651 EC50 = 17.57 nM T40474 COG79Z 86566652 EC50 = 17.53 nM T40474 CI4Y8R 86566672 EC50 = 27.91 nM T40474 CKYH94 86566673 EC50 = 12.37 nM T40474 C15RAH 86566674 EC50 = 81.24 nM T40474 CVUP97 86566675 EC50 = 24.59 nM T40474 CER02Z 86566677 EC50 = 39.96 nM T40474 C7E0AV 86566702 EC50 = 15.94 nM T40474 C6BGY4 86566796 IC50 = 2.04 nM T40474 C2TI1R 86566797 IC50 = 2.38 nM T40474 CR07OG 86566798 IC50 = 1.81 nM T40474 C08WGI 86566799 IC50 = 1.04 nM T40474 CE43DC 86566851 IC50 = 4.12 nM T40474 CH0Q2M 86567584 IC50 = 1.56 nM T40474 CDQN06 86567585 IC50 = 3.45 nM T40474 CKDR76 86567586 IC50 = 3.34 nM T40474 C6MG4E 86567587 IC50 = 2.13 nM T40474 C9HSM0 86567652 IC50 = 4.69 nM T40474 C96JYI 86567653 IC50 = 4.24 nM T40474 C36XYH 86567654 IC50 = 5.12 nM T40474 CZ3B7C 86567725 IC50 = 5.21 nM T40474 C9K3WP 86567726 IC50 = 4.35 nM T40474 C8N7GL 87123415 IC50 = 23 nM T40474 C3V6FU 87432100 IC50 = 16 nM T40474 C32VXS 87432117 IC50 = 3 nM T40474 C3Q0LD 87767734 IC50 = 5 nM T40474 CLE48M 89434293 IC50 = 9.9 nM T40474 C1HW4B 89735655 IC50 = 8500 nM T40474 CI5CD4 90267715 IC50 = 5800 nM T40474 C8Z1PB 90643473 IC50 = 165.5 nM T40474 CIMR30 90643474 IC50 = 70.2 nM T40474 CPAC09 90643475 IC50 = 100.8 nM T40474 CH5D1F 90643476 IC50 = 27 nM T40474 C6DWH1 90643477 IC50 = 290.5 nM T40474 C0HD4M 90643478 IC50 = 494.7 nM T40474 CD2Z9V 90643479 IC50 = 373.2 nM T40474 CGMS34 90643480 IC50 = 168.7 nM T40474 C6PW5H 90643481 IC50 = 49.6 nM T40474 CQL2G1 90643482 IC50 = 0.7 nM T40474 CB5O6E 90643483 IC50 = 1044 nM T40474 CC51BI 90643484 IC50 = 432.9 nM T40474 CR4KF8 90643485 IC50 = 427 nM T40474 CYX5U1 90643486 IC50 = 81 nM T40474 CHQX04 90643487 IC50 = 26.9 nM T40474 COR98Y 90644938 IC50 = 8.8 nM T40474 C07COR 90644939 IC50 = 7.9 nM T40474 CDZ5R6 90644940 IC50 = 32.5 nM T40474 CAP53K 90644941 IC50 = 66.4 nM T40474 CT9C6L 90644942 IC50 = 18.6 nM T40474 CWT52M 90644943 IC50 = 184 nM T40474 CUCN60 90644944 IC50 = 13.1 nM T40474 C7Z2LF 90644945 IC50 = 70.6 nM T40474 CM8JV5 90644946 IC50 = 337.6 nM T40474 C7K3FV 90644947 IC50 = 683.1 nM T40474 CNVW64 90644948 IC50 = 25.8 nM T40474 CY13SF 90644949 IC50 = 155.1 nM T40474 CAZO78 90644950 IC50 = 212.7 nM T40474 CQ71IN 90644951 IC50 = 234.3 nM T40474 CE3SB9 90644952 IC50 = 791.9 nM T40474 C9AS1Y 90644954 IC50 = 44.8 nM T40474 CQ5I8Z 90644955 IC50 = 23.4 nM T40474 C4DY8K 90644956 IC50 = 149.9 nM T40474 CD52AH 90644957 IC50 = 68.3 nM T40474 CHV49F 90644958 IC50 = 51.7 nM T40474 C6T9IR 90644959 IC50 = 113.8 nM T40474 C8GH1V 90644960 IC50 = 52.6 nM T40474 CXO2R8 90644961 IC50 = 186.5 nM T40474 C4IO7C 90644963 IC50 = 248.9 nM T40474 CJ21KA 90644964 IC50 = 21.7 nM T40474 C8F3XR 90644965 IC50 = 3.8 nM T40474 C6F9ET 90644966 IC50 = 81.9 nM T40474 C74CUT 90644967 IC50 = 104.9 nM T40474 CS36RL 90644968 IC50 = 643.1 nM T40474 C7QUR0 90644969 IC50 = 168.9 nM T40474 CWF9A4 90644970 IC50 = 924 nM T40474 CKI20G 90644971 IC50 = 805.8 nM T40474 CI2QL1 90644972 IC50 = 211.1 nM T40474 C5S3YB 90645165 IC50 = 2.15 nM T40474 CTS79Y 90645166 IC50 = 9.95 nM T40474 C68BJV 90645167 IC50 = 5.02 nM T40474 CC8BA1 90645168 IC50 = 5.63 nM T40474 C5AK8S 90645169 IC50 = 8.27 nM T40474 CCLV30 90645170 IC50 = 9.16 nM T40474 CY0UC4 90645194 IC50 > 10000 nM T40474 CK4G1F 90646071 IC50 = 8.34 nM T40474 C6K2PH 90646431 IC50 = 3.98 nM T40474 C0S1HF 90655767 IC50 = 7 nM T40474 CW5ZR6 90655768 IC50 = 5 nM T40474 C51MOA 90655769 IC50 = 978 nM T40474 CZ6U5W 90655770 IC50 = 1719 nM T40474 C7P6FQ 90655771 IC50 = 564 nM T40474 CXA18Y 90655772 IC50 = 1048 nM T40474 C15GJU 90655773 IC50 = 1664 nM T40474 C25CWH 90655774 IC50 = 1225 nM T40474 CFRI21 90655775 IC50 = 2692 nM T40474 CAIL45 90655776 IC50 = 2708 nM T40474 CVYA67 90655777 IC50 = 2705 nM T40474 CHAQ83 90655778 IC50 = 2.8 nM T40474 CNB2K3 90655779 IC50 = 6.1 nM T40474 C3TM0S 90655780 IC50 = 6.5 nM T40474 C6V7KD 90655781 IC50 = 5.2 nM T40474 C7TS4O 90655782 IC50 = 710 nM T40474 CPW01E 90655783 IC50 = 33 nM T40474 C1G6QK 90655784 IC50 = 6.4 nM T40474 CV1S6R 90655785 IC50 = 1.9 nM T40474 CDWP34 90655786 IC50 > 1000 nM T40474 CKD16A 90655787 IC50 > 1000 nM T40474 C6EUD2 90655788 IC50 > 1000 nM T40474 CO28UJ 90655789 IC50 > 1000 nM T40474 CAU5K7 90655790 IC50 > 1000 nM T40474 C5NZ7A 90655791 IC50 > 1000 nM T40474 CGP7R9 90655792 IC50 = 31 nM T40474 C42VGQ 90655793 IC50 = 31 nM T40474 CM38BR 90655794 IC50 = 58 nM T40474 CGP3C6 90667419 IC50 = 5.1 nM T40474 CF6MO3 90667420 IC50 = 1.2 nM T40474 CCO96L 90667421 IC50 = 1.2 nM T40474 C6ULI7 90667422 IC50 = 1.6 nM T40474 CIW51L 90667423 IC50 = 2.3 nM T40474 CG2J7Y 90667424 IC50 = 2.6 nM T40474 CC7G4Q 90667584 IC50 = 2.1 nM T40474 CW5UZ9 90667585 IC50 = 1.7 nM T40474 CGX4S0 90667586 IC50 = 5.1 nM T40474 C9XVG4 90667588 IC50 = 23.3 nM T40474 C08COA 90667590 IC50 = 155 nM T40474 C7A9YC 90667592 IC50 = 646 nM T40474 C7K2SL 90667593 IC50 = 324 nM T40474 CO29CA 90667598 IC50 = 146 nM T40474 CD01RM 90667599 IC50 = 235 nM T40474 C7BK1O 90667600 IC50 = 467 nM T40474 CF4WI1 90667601 IC50 = 263 nM T40474 CZL03G 90667602 IC50 = 3.9 nM T40474 CR59JY 90667603 IC50 = 254 nM T40474 CC5G2D 90667606 IC50 = 207 nM T40474 CGRK73 90667608 IC50 = 0.9 nM T40474 C2ZN9Y 90667609 IC50 = 1.6 nM T40474 CT5H7A 90667610 IC50 = 3 nM T40474 CTD7C6 90667611 IC50 = 0.7 nM T40474 C26KEM 91262312 IC50 = 10 nM T40474 C0Y8ZK 91933875 IC50 > 100 nM T40474 CAU45T 91971978 IC50 > 30000 nM T40474 C8F7XO 92131166 IC50 = 2.27 nM T40474 CZK0S7 101393982 IC50 > 20000 nM T40474 C6D9CA 101896448 IC50 = 5.2 nM T40474 C2VFS6 101898750 IC50 = 50 nM T40474 CK72FW 102129497 IC50 = 1.63 nM T40474 C34SPQ 102369824 IC50 = 7600 nM T40474 C08MIB 118705809 IC50 = 13.57 nM T40474 C0H7MN 118705810 IC50 = 4.31 nM T40474 CQR19I 118705811 IC50 = 3.98 nM T40474 CS5JE2 118705817 IC50 = 1.98 nM T40474 C7QW4N 118705941 IC50 = 2.03 nM T40474 CY7BI2 118706214 IC50 > 10000 nM T40474 C1RO4V 118709802 IC50 = 1340 nM T40474 CUD8S3 118709803 IC50 > 10000 nM T40474 CZ0NL4 118709804 IC50 = 8800 nM T40474 C2ZYH1 118709805 IC50 = 4540 nM T40474 C46SBZ 118709806 IC50 > 10000 nM T40474 CPE61B 118709808 IC50 = 7300 nM T40474 C3U5XI 118709809 IC50 = 7480 nM T40474 CV8Z3F 118709810 IC50 = 1500 nM T40474 CGT82L 118709811 IC50 > 10000 nM T40474 C4INY8 118709812 IC50 = 4240 nM T40474 CHR4E5 118709813 IC50 = 150 nM T40474 C6P4YN 118709814 IC50 = 560 nM T40474 C0FU6Y 118709815 IC50 > 10000 nM T40474 CRT83K 118709816 IC50 > 10000 nM T40474 CX1TZ3 118709817 IC50 > 10000 nM T40474 C4H8VY 118709818 IC50 > 10000 nM T40474 CRVP89 118709819 IC50 = 1530 nM T40474 C12WRM 118709820 IC50 = 3580 nM T40474 CAS3B5 118709821 IC50 = 7850 nM T40474 C2IN3C 118710236 IC50 = 31.1 nM T40474 CF2YR1 118710237 IC50 = 10.6 nM T40474 CI28QB 118713249 IC50 = 20 nM T40474 C0AGP9 118713920 IC50 > 1000 nM T40474 CHF50O 118713921 IC50 = 7 nM T40474 CBD92A 118713922 IC50 = 6 nM T40474 CBKO25 118714682 IC50 = 720 nM T40474 CH6WB1 118714683 IC50 = 20 nM T40474 CD3Q1K 118714684 IC50 = 4 nM T40474 C6UZL4 118714685 IC50 = 21 nM T40474 CH37UM 118714686 IC50 = 13 nM T40474 C9D5KM 118714687 IC50 = 6 nM T40474 CL8MF1 118714688 IC50 = 4 nM T40474 C50IJG 118714689 IC50 = 10 nM T40474 CFE5H0 118714690 IC50 = 110 nM T40474 CGVX10 118715991 IC50 = 5.86 nM T40474 C8AQH4 118715993 IC50 = 4.95 nM T40474 CWO9B7 118715995 IC50 = 1.86 nM T40474 CV6L7F 118715999 IC50 = 3.05 nM T40474 CHR2J3 118717023 IC50 = 8.48 nM T40474 CS5LY8 118717024 IC50 = 8.91 nM T40474 CNGU59 118717025 IC50 = 3.68 nM T40474 C37CON 118717026 IC50 = 3.02 nM T40474 C9HTQ2 118717027 IC50 = 15.49 nM T40474 CCN2T7 118717028 IC50 = 10.21 nM T40474 C8I6LF 118717029 IC50 = 11.21 nM T40474 CVD5S4 118717030 IC50 = 3.98 nM T40474 CI2QU5 118717031 IC50 = 2.54 nM T40474 CRPU14 118717032 IC50 = 17.28 nM T40474 C94EMB 118717033 IC50 = 13.42 nM T40474 CDI8G5 118717034 IC50 = 12.89 nM T40474 C24YZX 118717035 IC50 = 3.12 nM T40474 CCY7E9 118717036 IC50 = 19.39 nM T40474 CNC73L 118717037 IC50 = 14.23 nM T40474 CM9LS1 118717038 IC50 = 14.49 nM T40474 C0AK5H 118717039 IC50 = 4.89 nM T40474 C2EPD5 118717040 IC50 = 3.25 nM T40474 CLY3S1 118717041 IC50 = 5.29 nM T40474 CAY0M7 118717042 IC50 = 5.02 nM T40474 CMC1X8 118717043 IC50 = 15.39 nM T40474 CPTE69 118717044 IC50 = 5.09 nM T40474 CO4J8I 118717045 IC50 = 2.47 nM T40474 CAFN71 118717046 IC50 = 25.43 nM T40474 C0IUS3 118721850 IC50 = 6.5 nM T40474 C1NZT3 118721851 IC50 = 7.1 nM T40474 C9IR6M 118721852 IC50 = 52.5 nM T40474 CA07OH 118722207 IC50 = 16.4 nM T40474 CZ93GF 118722208 IC50 = 7.5 nM T40474 CKM9F5 118722209 IC50 = 33.6 nM T40474 CJU8I4 118722210 IC50 = 119.8 nM T40474 CBXC83 118722211 IC50 = 51.4 nM T40474 C9JMP7 118722212 IC50 > 1000 nM T40474 C4IG8N 118722213 IC50 = 6.9 nM T40474 CM9B4L 118722214 IC50 = 137 nM T40474 CW3HP9 118722215 IC50 > 1000 nM T40474 COI93D 118722216 IC50 = 26.8 nM T40474 CFN94B 118722217 IC50 = 143 nM T40474 CHX3I0 118722218 IC50 = 43.1 nM T40474 C8TBS4 118722219 IC50 = 292 nM T40474 C8Q6ON 118722220 IC50 = 35.2 nM T40474 CB7G8S 118722221 IC50 > 1000 nM T40474 CTWA53 118722222 IC50 > 1000 nM T40474 C3BLR8 118722223 IC50 = 389 nM T40474 CWTY65 118722224 IC50 = 148 nM T40474 C1ROT4 118722225 IC50 = 31.7 nM T40474 CIC5R2 118722226 IC50 = 549 nM T40474 C8UTX5 118722227 IC50 = 130 nM T40474 CY9W0C 118722228 IC50 = 102 nM T40474 CU8KS3 118722229 IC50 = 338 nM T40474 CVC74S 118722230 IC50 = 164 nM T40474 C5WR9T 118722231 IC50 > 1000 nM T40474 CO9CG3 118722232 IC50 = 112 nM T40474 CEFM78 118722233 IC50 = 448 nM T40474 C9OXS4 118722234 IC50 = 244 nM T40474 C2Z3FV 118722235 IC50 = 634 nM T40474 CHQ19T 118722236 IC50 > 1000 nM T40474 C3KLI5 118723185 IC50 > 100000 nM T40474 CB6AQ9 118724098 IC50 = 26000 nM T40474 CNW20P 118724104 IC50 = 3900 nM T40474 CYLI89 118724106 IC50 = 12700 nM T40474 CSJI94 118724111 IC50 = 2000 nM T40474 CAG58K 118724398 IC50 = 3600 nM T40474 CK70YD 118724399 IC50 > 50000 nM T40474 CCTS47 118724401 IC50 = 2900 nM T40474 C2L7VZ 118724403 IC50 = 209000 nM T40474 CL48NP 118724404 IC50 = 19500 nM T40474 CLE04I 118724405 IC50 = 260000 nM T40474 CC7O3G 118724406 IC50 = 20200 nM T40474 CV62QN 118726097 IC50 = 17.4 nM T40474 CJTV10 118726098 IC50 > 1000 nM T40474 CPR3Z7 118726099 IC50 > 1000 nM T40474 CG23FX 118726100 IC50 = 6.7 nM T40474 C4ZL9Y 118726101 IC50 = 566 nM T40474 C64STK 118726102 IC50 = 57.5 nM T40474 CB85CA 118726103 IC50 = 19.5 nM T40474 CY0GB4 118726104 IC50 = 42.7 nM T40474 C5YFN8 118726105 IC50 = 76.2 nM T40474 C9QL8C 118726106 IC50 = 2.8 nM T40474 C0BN7O 118726107 IC50 > 1000 nM T40474 C2K4VT 118726108 IC50 = 199 nM T40474 C80BFS 118726109 IC50 > 1000 nM T40474 CIU74H 118726110 IC50 > 1000 nM T40474 CX59VL 118726111 IC50 > 1000 nM T40474 C2ID9Y 118726112 IC50 > 1000 nM T40474 CIU2C0 118726113 IC50 > 1000 nM T40474 C5LN0H 118726114 IC50 = 138 nM T40474 CTR9K0 118726115 IC50 = 561 nM T40474 C0CLE5 118726116 IC50 > 1000 nM T40474 C82YOM 118726117 IC50 > 1000 nM T40474 CHT6K9 118728811 Ki > 4000 nM T40474 CUA3Y2 118728812 Ki > 4000 nM T40474 CDQ78G 118728813 Ki > 4000 nM T40474 CZ6XL7 118728814 Ki > 4000 nM T40474 CMO67K 118728815 Ki > 4000 nM T40474 CR2M0Q 118728816 Ki > 4000 nM T40474 C62SCL 118728817 Ki > 4000 nM T40474 CSB30C 118728819 Ki > 4000 nM T40474 CV7XU8 118728820 Ki > 4000 nM T40474 C3J1EX 118728821 Ki > 4000 nM T40474 CIWB78 118728822 Ki > 4000 nM T40474 CP18SE 118728823 Ki > 4000 nM T40474 CM42CA 118728824 Ki > 4000 nM T40474 C9Q7CL 118728825 Ki > 4000 nM T40474 CCR3S0 118728826 Ki > 4000 nM T40474 CD1H2L 118729329 IC50 = 300 nM T40474 C31DZN 118729330 IC50 = 200 nM T40474 CFU41Z 118732796 IC50 = 23 nM T40474 CCPQ28 118732797 IC50 = 32 nM T40474 CPYQ82 118732798 IC50 = 11 nM T40474 CR0W1T 118732799 IC50 = 7 nM T40474 CI2PT1 118732800 IC50 = 24 nM T40474 C8BF6A 118732801 IC50 = 18 nM T40474 CR4JB0 118732802 IC50 = 11 nM T40474 COPN74 118732803 IC50 = 182 nM T40474 CIX08G 118732804 IC50 = 67 nM T40474 C4ZX7Y 118732957 IC50 = 52 nM T40474 C8HFD1 118732958 IC50 = 4 nM T40474 CAY5J3 118732959 IC50 = 2 nM T40474 CM4NV8 118732960 IC50 = 7 nM T40474 CXG02Y 118732961 IC50 = 1 nM T40474 C7R8HJ 118732962 IC50 = 1 nM T40474 C53QIC 118732963 IC50 > 400 nM T40474 CW79TK 118732964 IC50 = 93 nM T40474 CK3S7W 118732965 IC50 = 67 nM T40474 CWT64X 118734826 IC50 = 370 nM T40474 CTH03L 118734827 IC50 = 46 nM T40474 CYHZ19 118734828 IC50 = 191 nM T40474 C9BQI8 118734829 IC50 = 39.5 nM T40474 C70PKI 118734830 IC50 = 17 nM T40474 C16JVK 118734831 IC50 = 51 nM T40474 CH7ZJ4 118734832 IC50 = 24 nM T40474 C0NJ8G 118734833 IC50 = 19 nM T40474 CF5C3S 118734834 IC50 = 20 nM T40474 CSE0N6 118734835 IC50 = 36 nM T40474 C19ALQ 118734836 IC50 = 9 nM T40474 CJQR31 118734837 IC50 = 10 nM T40474 C31CFI 118734838 IC50 = 2.3 nM T40474 C3EBP6 118734839 IC50 = 1.7 nM T40474 CR25IU 118734840 IC50 = 9.8 nM T40474 CF7MI1 118734841 IC50 = 5.2 nM T40474 CUB64A 118734842 IC50 = 10.7 nM T40474 CZT16K 118734843 IC50 = 10000 nM T40474 CEZ91Y 118734844 IC50 > 10000 nM T40474 CA07SM 118734845 IC50 > 10000 nM T40474 CDF95U 118734846 IC50 = 190 nM T40474 CRY5E8 118734847 IC50 = 320 nM T40474 C4V6QD 118734848 IC50 = 89 nM T40474 C2TAE6 118935328 IC50 > 1000 nM T40474 C2TF6E 122179286 IC50 = 2400 nM T40474 CM04OW 122179287 IC50 = 670 nM T40474 C4YR9I 122179288 IC50 = 3770 nM T40474 CJ76AF 122179289 IC50 = 4370 nM T40474 C1T7CU 122179290 IC50 = 5780 nM T40474 C9PC2V 122179432 IC50 = 3.2 nM T40474 CBO8R5 122179433 IC50 = 4.3 nM T40474 CC0FY5 122179434 IC50 = 5.6 nM T40474 C21VAG 122179435 IC50 = 14.5 nM T40474 CM6LW0 122179436 IC50 = 3.3 nM T40474 C4RPI6 122179437 IC50 = 2.8 nM T40474 C7GZB4 122179438 IC50 = 9.7 nM T40474 CK9X5I 122179439 IC50 = 16.2 nM T40474 CT12KS 122179440 IC50 = 12.8 nM T40474 CO1ZF6 122179441 IC50 = 10.6 nM T40474 CY6C1E 122179442 IC50 = 3.9 nM T40474 C5XR0O 122179443 IC50 = 8.3 nM T40474 CRLF62 122179444 IC50 = 4.7 nM T40474 CXZ73K 122179445 IC50 = 0.13 nM T40474 C08KEM 122179540 IC50 = 5100 nM T40474 C3AJ4C 122179546 IC50 = 7700 nM T40474 CG0RP7 122179547 IC50 = 4300 nM T40474 C1A0SQ 122179548 IC50 = 5700 nM T40474 CT1PU6 122182086 IC50 = 35.68 nM T40474 C6ZRP0 122182088 IC50 = 31.2 nM T40474 CWF23H 122182089 IC50 = 28.54 nM T40474 C9EGL0 122182090 IC50 = 23.86 nM T40474 CF8ED9 122182092 IC50 = 24.25 nM T40474 CSE7Q3 122182094 IC50 = 27.3 nM T40474 C30VQU 122182095 IC50 = 6.26 nM T40474 CL17OK 122182096 IC50 = 5.41 nM T40474 CQ1FL4 122182097 IC50 = 5.64 nM T40474 C4B7XO 122182098 IC50 = 4.36 nM T40474 CID02H 122182232 IC50 = 18.44 nM T40474 CPI79H 122182233 IC50 = 13.3 nM T40474 CU41TZ 122182234 IC50 = 18.6 nM T40474 C6CLO3 122182235 IC50 = 7.43 nM T40474 CJ13HZ 122182236 IC50 = 5.8 nM T40474 C93FVA 122182237 IC50 = 6.67 nM T40474 C63PDV 122182238 IC50 = 5.16 nM T40474 CV48EB 122182239 IC50 = 25.49 nM T40474 C54BVL 122182240 IC50 = 20.54 nM T40474 CAD89F 122182241 IC50 = 14.68 nM T40474 C8CF5L 122182402 IC50 = 10.64 nM T40474 C2TGE5 122182403 IC50 = 26.18 nM T40474 C0CRY8 122182404 IC50 = 19.22 nM T40474 CY14RM 122182405 IC50 = 10.86 nM T40474 C2QV6H 122182406 IC50 = 8.1 nM T40474 CW6D3J 122182407 IC50 = 4.16 nM T40474 C98SBG 122182408 IC50 = 2.9 nM T40474 CWA94G 122182409 IC50 = 1.42 nM T40474 C9OWX5 122186256 IC50 > 10000 nM T40474 C3J6BA 122186261 IC50 > 10000 nM T40474 C53FOD 122186955 IC50 = 740 nM T40474 CGB2M4 122186956 IC50 = 2070 nM T40474 C3DQG0 122186957 IC50 = 2260 nM T40474 C2QP6A 122186958 IC50 = 4840 nM T40474 CYA03Q 122186959 IC50 = 1090 nM T40474 CP3M2E 122186960 IC50 = 350 nM T40474 CHL1E7 122186961 IC50 = 1230 nM T40474 CK48SW 122186962 IC50 = 7 nM T40474 C4GIB5 122186963 IC50 = 10 nM T40474 C3EH6R 122186964 IC50 = 190 nM T40474 CZE7O3 122187075 IC50 > 10000 nM T40474 C4JC0N 122187076 IC50 > 10000 nM T40474 CW7K4G 122187077 IC50 = 340 nM T40474 C1R8VS 122187846 IC50 = 304 nM T40474 C3X8BL 122187848 IC50 = 108 nM T40474 CPC26B 122187849 IC50 = 58 nM T40474 CZN2V0 122188510 IC50 = 2427 nM T40474 C4X7SD 122192466 IC50 > 10000 nM T40474 CNX0Q2 122193763 IC50 > 10000 nM T40474 CWV0C3 122193764 IC50 > 10000 nM T40474 CSG98Y 122193765 IC50 > 10000 nM T40474 CCLQ75 122193769 IC50 > 10000 nM T40474 CXDR48 122193770 IC50 > 10000 nM T40474 CPA8C5 122193773 IC50 > 10000 nM T40474 CBT9C4 123372252 IC50 = 5.3 nM T40474 C4SDK1 127025214 IC50 = 12.2 nM T40474 CS4PU5 127025215 IC50 = 20.1 nM T40474 C7UH9I 127025216 IC50 = 4.3 nM T40474 CLTA86 127025515 IC50 = 5.6 nM T40474 C1WB2U 127025516 IC50 = 7.3 nM T40474 C3FVQ2 127025839 IC50 > 100 nM T40474 C3BX9T 127025840 IC50 > 100 nM T40474 C4WVZ8 127025841 IC50 = 82.1 nM T40474 C9VX3I 127025842 IC50 > 100 nM T40474 C8KXV1 127025843 IC50 = 7.5 nM T40474 CR2TG8 127025844 IC50 = 8.1 nM T40474 C0H6JF 127026113 IC50 = 27.9 nM T40474 CGXD47 127026114 IC50 = 10.5 nM T40474 CKX3Y1 127026115 IC50 = 53.2 nM T40474 C7VS2I 127026118 IC50 = 15.9 nM T40474 C01MEW 127026130 IC50 > 100 nM T40474 C5M9HV 127026174 IC50 = 62.82 nM T40474 CRZ0E7 127026178 IC50 = 8.92 nM T40474 CJZT69 127026430 IC50 = 3.6 nM T40474 C18KQJ 127026431 IC50 = 15.9 nM T40474 C2MQZ6 127026487 IC50 = 121.42 nM T40474 CRVO69 127026524 IC50 = 72.33 nM T40474 CYA7E0 127026527 IC50 = 13.51 nM T40474 CDJE19 127027007 IC50 = 21.2 nM T40474 CCW8P7 127027081 IC50 = 4.3 nM T40474 C8LPN4 127027082 IC50 = 18.8 nM T40474 C2TH4S 127027083 IC50 > 100 nM T40474 CUV84M 127027331 IC50 = 13.6 nM T40474 CV76EN 127027385 IC50 > 100 nM T40474 CEG0W4 127027437 IC50 = 56.42 nM T40474 CB53ZX 127028515 IC50 > 10000 nM T40474 CB9VY8 127028516 IC50 > 10000 nM T40474 CAD38Y 127029440 IC50 > 10000 nM T40474 CR17GV 127029715 IC50 > 10000 nM T40474 C1XD6R 127029809 IC50 = 1.21 nM T40474 C1ZM6U 127029862 IC50 = 42.56 nM T40474 CZ9B6S 127029863 IC50 = 5.24 nM T40474 CI1E5W 127029864 IC50 = 1.68 nM T40474 CRX3A4 127030383 IC50 = 11 nM T40474 CTX1I0 127030562 IC50 = 29.27 nM T40474 C7QE5U 127030563 IC50 = 37.71 nM T40474 C8QCK0 127030564 IC50 = 19.36 nM T40474 C5MPB4 127030789 IC50 = 12.18 nM T40474 CMQ03C 127030818 IC50 = 7.25 nM T40474 C8CSR2 127030860 IC50 = 16.25 nM T40474 CJW0U8 127030861 IC50 = 14.74 nM T40474 C43NUR 127030862 IC50 = 25.42 nM T40474 COQ6Y2 127030935 IC50 = 6 nM T40474 CV3M9G 127030954 IC50 = 15.7 nM T40474 CCD4B3 127031098 IC50 = 5.32 nM T40474 CMF6X9 127031103 IC50 = 12.51 nM T40474 C9WG2J 127031106 IC50 = 18.39 nM T40474 C7CZ5I 127031145 IC50 = 10.73 nM T40474 CK36YE 127031146 IC50 = 6.39 nM T40474 COTG01 127031447 IC50 = 16.38 nM T40474 CXGJ91 127031448 IC50 = 21.27 nM T40474 C4D2NL 127031449 IC50 = 19.39 nM T40474 CP3R1O 127031480 IC50 = 980 nM T40474 C15CWS 127031933 IC50 = 3.8 nM T40474 C15RAX 127031934 IC50 = 47.8 nM T40474 C7RUK3 127031935 IC50 = 5.6 nM T40474 C6TUY3 127031936 IC50 = 18.9 nM T40474 CL15BU 127031937 IC50 < 10 nM T40474 CZN21Y 127032011 IC50 = 3400 nM T40474 C5DVO6 127032056 IC50 = 16.82 nM T40474 CERB36 127032057 IC50 = 14.34 nM T40474 C7XOL0 127032058 IC50 = 12.78 nM T40474 CBA64T 127032059 IC50 = 24.14 nM T40474 C64IPH 127032060 IC50 = 21.63 nM T40474 CM9J6I 127032205 IC50 = 3.8 nM T40474 C9QK2Y 127032206 IC50 = 11 nM T40474 C2QK3P 127032207 IC50 = 3.4 nM T40474 C62GEC 127032332 IC50 = 12.56 nM T40474 CPC73Y 127032638 IC50 = 11.26 nM T40474 C0GSE8 127032639 IC50 = 15.69 nM T40474 CH03QK 127032640 IC50 = 18.15 nM T40474 CJM5L9 127032641 IC50 = 11.37 nM T40474 CS1LC4 127032678 IC50 = 2200 nM T40474 C5FIL6 127033117 IC50 = 19.5 nM T40474 C7W3AL 127033393 IC50 = 42.3 nM T40474 C63JFM 127033394 IC50 = 105.1 nM T40474 CM3Z1Y 127033395 IC50 = 33.5 nM T40474 CO8QE6 127033396 IC50 = 93.6 nM T40474 CUH79P 127033397 IC50 = 9.8 nM T40474 CZG6F5 127033774 IC50 = 6.84 nM T40474 CRF0C1 127034162 IC50 = 120 nM T40474 CYK8U5 127034321 IC50 = 3.26 nM T40474 CDU62W 127034324 IC50 = 1.75 nM T40474 C8T0KB 127034388 IC50 = 21.49 nM T40474 CV8CF0 127034389 IC50 = 22.33 nM T40474 CLH45I 127034396 IC50 = 21.26 nM T40474 C9UQY1 127034548 IC50 = 7.6 nM T40474 C85VMN 127034549 IC50 = 3.5 nM T40474 C2F3RC 127034550 IC50 = 5.9 nM T40474 C54HFT 127034551 IC50 = 5.1 nM T40474 CR4JX6 127034553 IC50 = 1 nM T40474 CKS28E 127034802 IC50 > 1000 nM T40474 C1APH7 127036195 IC50 > 10000 nM T40474 CE3QV2 127036196 IC50 = 7300 nM T40474 COG5C4 127036197 IC50 = 8200 nM T40474 CVP5G9 127036198 IC50 > 10000 nM T40474 C3K7HL 127036199 IC50 > 10000 nM T40474 C8V5FX 127036375 IC50 > 10000 nM T40474 CPF19C 127036376 IC50 = 6600 nM T40474 C9E2LI 127036377 IC50 > 10000 nM T40474 CI25YV 127036378 IC50 > 10000 nM T40474 CO9XA5 127036379 IC50 = 8900 nM T40474 CQ7EJ1 127036407 IC50 = 5900 nM T40474 C27NGV 127036408 IC50 > 10000 nM T40474 C63QEV 127036409 IC50 = 610 nM T40474 CQX54Z 127036431 IC50 = 690 nM T40474 CGHD79 127036567 IC50 = 2200 nM T40474 C3IQ7U 127036568 IC50 > 10000 nM T40474 CFVN61 127036569 IC50 > 10000 nM T40474 CNQ45A 127037197 IC50 = 2300 nM T40474 CQ3M5O 127037198 IC50 = 1600 nM T40474 C0YW6O 127037199 IC50 > 10000 nM T40474 CB6I1A 127037200 IC50 = 4600 nM T40474 CZL2S7 127037243 IC50 = 5230 nM T40474 CM0DX3 127037244 IC50 = 890 nM T40474 CXYW65 127037245 IC50 = 1210 nM T40474 C8TB3R 127041351 IC50 = 1 nM T40474 C40WEH 127041352 IC50 > 1.8 nM T40474 C8ZUW1 127042632 IC50 = 54.25 nM T40474 C8M9GK 127042961 IC50 = 15.67 nM T40474 CYC39L 127043322 IC50 = 3630 nM T40474 C5SIW0 127043323 IC50 = 2600 nM T40474 CEJD06 127043499 IC50 = 4880 nM T40474 CY72HU 127043769 IC50 = 11770 nM T40474 CI1SW6 127044032 IC50 = 11780 nM T40474 C5SJN7 127044033 IC50 = 18900 nM T40474 CR3BC7 127044034 IC50 = 4010 nM T40474 CJ71RB 127044431 IC50 = 7900 nM T40474 CA8EF4 127044577 IC50 = 6 nM T40474 CK1AS9 127044693 IC50 = 23700 nM T40474 CTQJ69 127045456 IC50 = 6730 nM T40474 CJG1R7 127045457 IC50 = 11990 nM T40474 C3XA8K 127045458 IC50 = 7600 nM T40474 C3MP0W 127045459 IC50 > 20000 nM T40474 C8ERJ7 127045762 IC50 = 0.24 nM T40474 CX4CJ5 127045832 IC50 = 0.5 nM T40474 C1D0XF 127045833 IC50 = 0.67 nM T40474 CHK16Q 127045929 IC50 > 1000 nM T40474 CX9U8E 127046394 IC50 = 0.42 nM T40474 CW62RS 127046732 IC50 = 0.59 nM T40474 CY3J0C 127047591 IC50 > 1000 nM T40474 C4I0EL 127048223 IC50 = 5200 nM T40474 CP4I1C 127048227 IC50 = 6900 nM T40474 C1LGA8 127048248 IC50 = 2300 nM T40474 CI0Q8P 127048249 IC50 = 3200 nM T40474 CA41FB 127048250 IC50 = 3500 nM T40474 CYD1I7 127048271 IC50 = 5300 nM T40474 C9F1CL 127048332 IC50 = 980 nM T40474 CI30SM 127048567 IC50 = 1100 nM T40474 C28RKY 127049237 IC50 = 5800 nM T40474 CR9C5O 127049568 IC50 > 20000 nM T40474 CO69DV 127049906 IC50 = 12200 nM T40474 CE0RI5 127050089 IC50 = 8.75 nM T40474 CZI86H 127050090 IC50 > 20000 nM T40474 C0V1UO 127050091 IC50 > 20000 nM T40474 CWO8P5 127050092 IC50 > 20000 nM T40474 C58JVE 127050200 IC50 > 20000 nM T40474 COC17T 127050404 IC50 = 8200 nM T40474 C2M0GE 127050496 IC50 = 8500 nM T40474 C8TEC9 127050825 IC50 = 1300 nM T40474 C9T8XM 127051082 IC50 = 1200 nM T40474 CXTD47 127051095 IC50 = 3.08 nM T40474 C9X3RD 127051099 IC50 = 11400 nM T40474 C50YIT 127051394 IC50 = 8300 nM T40474 CX0V6S 127051395 IC50 = 1200 nM T40474 C7ZV9H 127051396 IC50 = 8000 nM T40474 CV60KL 127051407 IC50 = 6.68 nM T40474 CNWF24 127052031 IC50 > 20000 nM T40474 CA97MR 127052127 IC50 = 420 nM T40474 CF2S6N 127052258 IC50 = 5200 nM T40474 C7TNW0 127052339 IC50 = 9100 nM T40474 CRU8M3 127052561 IC50 = 1000 nM T40474 CYQP42 127052562 IC50 = 6100 nM T40474 CSM06R 127052848 IC50 > 20000 nM T40474 CW4H6O 127052849 IC50 > 20000 nM T40474 CJHE94 127052850 IC50 > 20000 nM T40474 C9RM1X 127052851 IC50 > 20000 nM T40474 CB7X4E 127052852 IC50 > 20000 nM T40474 CJ3NT4 127052949 IC50 > 20000 nM T40474 C2XV0E 127053159 IC50 = 9.45 nM T40474 CVMC24 127053160 IC50 = 10.37 nM T40474 C9Q8ZR 127053161 IC50 > 20000 nM T40474 CY3CF2 127053162 IC50 = 2100 nM T40474 CUO0C5 132156633 IC50 > 10000 nM T40474 C53OJM 132607333 IC50 = 0.9 nM T40474 CRK91M 132607334 IC50 = 2.35 nM T40474 CX3SA0 132607335 IC50 = 1.22 nM T40474 C3HO4V 132819884 IC50 = 43 nM T40474 C94TWB 132819885 IC50 = 3.9 nM T40474 CYT5G2 132819886 IC50 = 63 nM T40474 C9CBE0 132819887 IC50 = 20 nM T40474 CMI3Q0 132819888 IC50 = 1.1 nM T40474 CSXT74 132819889 IC50 = 21 nM T40474 CA04HJ 132819891 IC50 = 58 nM T40474 CJ45WS 132819892 IC50 = 17 nM T40474 CA0M5D 132819893 IC50 = 5.6 nM T40474 CM8XS4 132819894 IC50 = 35 nM T40474 CERS64 132937256 EC50 = 1.45 nM T40474 CX9E3P 134132094 IC50 = 4.33 nM T40474 CN6IW4 134132401 IC50 = 31 nM T40474 CL5JT8 134132828 IC50 = 3.85 nM T40474 CVO3Q0 134133897 IC50 = 106.4 nM T40474 CPJG85 134135151 IC50 = 376 nM T40474 C0GFR4 134136001 IC50 = 19 nM T40474 C9FZ3A 134136788 IC50 = 157 nM T40474 CG92RQ 134137314 IC50 = 380 nM T40474 CURF53 134137336 IC50 = 51.6 nM T40474 CQ3YV8 134137418 IC50 = 46.5 nM T40474 C7I5FB 134137427 IC50 = 22 nM T40474 C1U2MV 134137679 IC50 = 479 nM T40474 CH42QO 134138567 IC50 = 29 nM T40474 C6FZ9M 134139131 IC50 = 3.03 nM T40474 CHL7B1 134140023 IC50 > 1000 nM T40474 CHIN70 134140111 IC50 = 103.2 nM T40474 C6M9DN 134140179 IC50 = 220 nM T40474 C8KC5F 134142230 IC50 = 393 nM T40474 C8VL1A 134144165 IC50 = 13.08 nM T40474 CEBA68 134144540 IC50 = 8.66 nM T40474 CYK69E 134145349 IC50 = 37.5 nM T40474 CQ71TG 134145719 IC50 = 84.6 nM T40474 CETL92 134145932 IC50 = 18 nM T40474 CU20AE 134146499 IC50 = 47.5 nM T40474 CGE8X4 134146851 IC50 = 56.3 nM T40474 CJUY81 134146873 IC50 = 2.08 nM T40474 CHZT39 134147040 IC50 = 10.15 nM T40474 CRM5C8 134147151 IC50 = 89.8 nM T40474 CMJ6X4 134147909 IC50 = 31.52 nM T40474 CUKE45 134147919 IC50 = 1.57 nM T40474 CDCJ80 134148182 IC50 > 1000 nM T40474 C7S2XA 134148711 IC50 = 11.15 nM T40474 CN0X6S 134149608 IC50 = 4.55 nM T40474 C08NSE 134151557 IC50 = 8.2 nM T40474 CJK46H 134152689 IC50 = 9.9 nM T40474 C3IO8Y 134154183 IC50 = 89.3 nM T40474 CS52QP 134155152 IC50 = 24 nM T40474 C6TUP1 134156489 IC50 = 17.3 nM T40474 CVGT85 134158009 IC50 = 53.1 nM T40474 C2AN7T 134611886 IC50 > 100000 nM T40474 CZ8W6R 134612705 IC50 > 1000 nM T40474 CYL5V1 134694986 IC50 = 0.48 nM T40474 CKH4M7 135407905 IC50 = 5 nM T40474 CV3Z7D 135407907 IC50 = 100 nM T40474 CH0TR1 135407908 IC50 = 5 nM T40474 C42BQM 135407909 IC50 = 0.7 nM T40474 C6ZHV5 135407910 IC50 = 0.5 nM T40474 CK8ML6 135407911 IC50 = 2 nM T40474 C3CDT7 135407912 IC50 = 1.6 nM T40474 CMP71Q 135407919 IC50 = 10 nM T40474 CX6VT0 135407920 IC50 = 1 nM T40474 CFH34T 135440116 IC50 = 12 nM T40474 CWRI46 135475228 IC50 = 7038 nM T40474 CJ4AP0 135481052 IC50 = 7 nM T40474 C84SAN 135511699 IC50 = 489 nM T40474 CJI0G1 135520135 IC50 > 10000 nM T40474 CTJ48K 135524085 IC50 = 140 nM T40474 CUT1W7 135524168 IC50 = 85 nM T40474 CEUW05 135537650 IC50 = 7 nM T40474 CE8MF0 135566634 Ki = 1.3 nM T40474 C23VIF 135653162 IC50 = 79.3 nM T40474 CPV59N 135685787 Ki > 4000 nM T40474 C29PWN 135886762 IC50 > 50000 nM T40474 CF1PS8 135934877 Ki > 4000 nM T40474 CTRL59 135976660 Ki > 4000 nM T40474 CHA4N2 136013680 IC50 > 10 nM T40474 C61VJS 136025823 IC50 = 65 nM T40474 C8C3QA 136025875 IC50 = 43 nM T40474 C7SJ5E 136025883 IC50 = 22 nM T40474 C2IEF4 136025884 IC50 = 90 nM T40474 C6KXU0 136025885 IC50 = 59 nM T40474 C5EV9N 136025905 IC50 = 58 nM T40474 CVN43Z 136025906 IC50 = 320 nM T40474 C0TNH3 136025907 IC50 = 29 nM T40474 CE28BU 136025908 IC50 = 1300 nM T40474 CF6K8B 136025909 IC50 = 3100 nM T40474 CC6DV1 136026016 IC50 = 23 nM T40474 C9M2HF 136026017 IC50 = 230 nM T40474 CCP7F9 136026018 IC50 = 46 nM T40474 C6ZLI2 136026032 IC50 = 13 nM T40474 CUC4A5 136026033 IC50 = 1770 nM T40474 C1NMQ0 136026034 IC50 = 630 nM T40474 CVMW43 136026035 IC50 = 5990 nM T40474 C0J8TO 136026036 IC50 = 420 nM T40474 CT36OP 136026053 IC50 = 130 nM T40474 C2VU1O 136026054 IC50 = 5840 nM T40474 CIQV96 136026055 IC50 = 230 nM T40474 CUB58F 136026056 IC50 = 980 nM T40474 C6IE4W 136026057 IC50 = 7200 nM T40474 C27QJO 136026058 IC50 = 520 nM T40474 C12NSM 136026078 IC50 = 1620 nM T40474 C6T9GI 136026171 IC50 = 570 nM T40474 CBQ37F 136026172 IC50 = 29 nM T40474 CF47WZ 136026173 IC50 = 16 nM T40474 CO4BW9 136026174 IC50 = 20 nM T40474 CVCH89 136026183 IC50 = 1450 nM T40474 C0WFQ3 136026184 IC50 = 37 nM T40474 C04MCP 136026185 IC50 = 65 nM T40474 CT28DQ 136026186 IC50 = 20 nM T40474 CF3MJ0 136026187 IC50 = 170 nM T40474 CQ4TG6 136026188 IC50 = 15 nM T40474 CJ8G7T 136026189 IC50 = 89 nM T40474 CF64PM 136026190 IC50 = 3340 nM T40474 C4L5ZJ 136026191 IC50 = 200 nM T40474 CRD1I7 136042199 IC50 = 5 nM T40474 CJ7U4C 136053657 IC50 = 1.54 nM T40474 C6STL8 136068598 IC50 = 200 nM T40474 C1ZFE4 136068599 IC50 = 16 nM T40474 CKI91Q 136068604 IC50 = 15 nM T40474 C24ZHI 136068605 IC50 = 21 nM T40474 CI6AH4 136068626 IC50 = 65 nM T40474 CGTO72 136068627 IC50 = 900 nM T40474 C3PEG6 136068628 IC50 = 1060 nM T40474 C3TE9B 136068629 IC50 = 500 nM T40474 C7SUP9 136068630 IC50 = 890 nM T40474 CYMA74 136068631 IC50 = 24 nM T40474 C68SPH 136068709 IC50 = 1 nM T40474 C42OAU 136068710 IC50 = 140 nM T40474 CV9A0H 136068711 IC50 = 2150 nM T40474 CW1G8Y 136086942 IC50 = 21 nM T40474 CXI5Q1 136086943 IC50 = 36 nM T40474 CRPW29 136086944 IC50 = 13 nM T40474 C7WSE8 136086945 IC50 = 81 nM T40474 CW8V2Z 136086946 IC50 = 32 nM T40474 CX65ZL 136086947 IC50 = 54 nM T40474 C5PUI2 136086948 IC50 = 55 nM T40474 C04VFZ 136086949 IC50 = 91 nM T40474 CYZ23A 136086950 IC50 = 2000 nM T40474 C4V0NG 136086951 IC50 = 3080 nM T40474 C9S2UJ 136086952 IC50 = 320 nM T40474 C6M9PF 136086953 IC50 = 45 nM T40474 C27WAP 136086954 IC50 = 190 nM T40474 CVD8Z7 136086955 IC50 = 180 nM T40474 CB9Q0U 136086956 IC50 = 790 nM T40474 CDT92U 136086957 IC50 = 2500 nM T40474 CRD7U0 136086958 IC50 = 47 nM T40474 C1B3CE 136086959 IC50 = 26 nM T40474 C9VUQ4 136086960 IC50 = 24 nM T40474 C0KM9X 136086961 IC50 = 8 nM T40474 CWT6N8 136086962 IC50 = 110 nM T40474 CKH84E 136086963 IC50 = 260 nM T40474 CY9VB3 136086964 IC50 = 24 nM T40474 CHF50Q 136086965 IC50 = 28 nM T40474 CSR4K5 136086966 IC50 = 0.7 nM T40474 C4NHP7 136086967 IC50 = 656 nM T40474 CU6N2Z 136086968 IC50 = 4700 nM T40474 CX52GJ 136086969 IC50 = 158 nM T40474 C7QPX5 136086970 IC50 = 78 nM T40474 C73TCA 136086971 IC50 = 430 nM T40474 CY8C9N 136086972 IC50 = 250 nM T40474 C3CAU4 136086973 IC50 = 150 nM T40474 C9JF6N 136086974 IC50 = 77 nM T40474 C0TIL9 136086975 IC50 = 78 nM T40474 CG1WD3 136086976 IC50 = 390 nM T40474 C0I8JN 136086977 IC50 = 86 nM T40474 CL6KD9 136086978 IC50 = 2080 nM T40474 CEC18P 136086979 IC50 = 4150 nM T40474 CH3E5A 136086980 IC50 = 110 nM T40474 CMC3S0 136086981 IC50 = 430 nM T40474 C4N2IC 136086982 IC50 = 5100 nM T40474 C0RT6Z 136086983 IC50 = 740 nM T40474 CF6NS1 136086984 IC50 = 5920 nM T40474 CJDT36 136086985 IC50 = 6160 nM T40474 CWP9X0 136086986 IC50 = 540 nM T40474 CNK81C 136086987 IC50 = 1050 nM T40474 CFJ84I 136086988 IC50 = 230 nM T40474 CN9T2G 136086989 IC50 = 30 nM T40474 CIX5Y9 136086990 IC50 = 6350 nM T40474 CJE92R 136086991 IC50 = 20 nM T40474 CA4EN3 136086992 IC50 = 15 nM T40474 CI96NU 136086993 IC50 = 54 nM T40474 C8CK2T 136086994 IC50 = 22 nM T40474 CD2W8C 136086995 IC50 = 240 nM T40474 CV5O1A 136086996 IC50 = 54 nM T40474 C1YB8O 136086997 IC50 = 110 nM T40474 C6D9BT 136086998 IC50 = 22 nM T40474 CAW79V 136086999 IC50 = 17 nM T40474 C7LFU6 136087000 IC50 = 210 nM T40474 CSEV18 136087001 IC50 = 67 nM T40474 CXST06 136087002 IC50 = 45 nM T40474 CW8JV4 136087003 IC50 = 88 nM T40474 CSHN51 136087004 IC50 = 1450 nM T40474 C0SZ5N 136087005 IC50 = 110 nM T40474 C95URZ 136087006 IC50 = 150 nM T40474 CT1H5F 136087007 IC50 = 6 nM T40474 CSKN65 136087008 IC50 = 1230 nM T40474 COP31J 136099320 IC50 = 9 nM T40474 CI28PO 136101243 IC50 > 20000 nM T40474 COC4N2 136101255 IC50 = 9 nM T40474 CAJ8N6 136101257 IC50 > 20000 nM T40474 C1UQL0 136101270 IC50 = 9 nM T40474 CW9K8Z 136126666 IC50 = 800 nM T40474 CH64ID 136175114 IC50 > 10000 nM T40474 CQ84IZ 136180335 Ki > 4000 nM T40474 CDT7E4 136211077 IC50 > 100 nM T40474 C9RE8D 136215817 IC50 = 1.15 nM T40474 CJX68G 136215836 IC50 = 4.31 nM T40474 CU53LY 136215837 IC50 = 2.58 nM T40474 CGSM70 136215838 IC50 = 3.72 nM T40474 C61LAJ 136215839 IC50 = 3.64 nM T40474 C14BIL 136215853 IC50 = 9.27 nM T40474 C7DIE6 136215854 IC50 = 3.15 nM T40474 CC9EP4 136215855 IC50 = 18.54 nM T40474 CT1WA4 136215864 IC50 = 3.84 nM T40474 CAE5L0 136215865 IC50 = 1.64 nM T40474 CLH95M 136215866 IC50 = 2.83 nM T40474 CJBL84 136215867 IC50 = 3.09 nM T40474 CFG48M 136215875 IC50 = 15.96 nM T40474 CVN9J2 136215876 IC50 = 4.82 nM T40474 C1T3JR 136215877 IC50 = 18.25 nM T40474 C15CHZ 136215885 IC50 = 3.36 nM T40474 C0JVH7 136215886 IC50 = 2.35 nM T40474 CST84N 136215887 IC50 = 2.68 nM T40474 CFP03J 136215888 IC50 = 12.39 nM T40474 CP9JC3 136215894 IC50 = 7.51 nM T40474 CPJ01L 136215895 IC50 = 2.38 nM T40474 C9SX1O 136215896 IC50 = 4.57 nM T40474 C9LQ1X 136215903 IC50 = 2.16 nM T40474 C6L4PW 136215904 IC50 = 3.03 nM T40474 C8OS6H 136215905 IC50 = 3.58 nM T40474 CQ2A7W 136215906 IC50 = 12.36 nM T40474 CSZ8C4 136216043 IC50 = 5.14 nM T40474 C8N7WO 136216044 IC50 = 21.24 nM T40474 CTHD14 136216045 IC50 = 3.29 nM T40474 C9J3PZ 136216063 IC50 = 2.68 nM T40474 C0EI2R 136216064 IC50 = 3.26 nM T40474 C5H4VW 136216065 IC50 = 3.15 nM T40474 CLP8B4 136216066 IC50 = 8.35 nM T40474 CDA84T 136216083 IC50 = 3.15 nM T40474 CL61YQ 136216084 IC50 = 8.14 nM T40474 CTBG70 136219238 IC50 = 330 nM T40474 C1YUD0 136219394 IC50 > 10 nM T40474 CXQL14 136239428 IC50 = 130 nM T40474 CKZ31H 136249503 IC50 = 140 nM T40474 C3WK7B 136249507 IC50 = 360 nM T40474 C8T9HP 136251282 IC50 = 89 nM T40474 CRV68G 136254210 IC50 = 8 nM T40474 CIU8W3 136254389 IC50 > 10 nM T40474 CW0FE9 137083622 IC50 > 10000 nM T40474 C4G5IA 137125270 IC50 = 207 nM T40474 CSGM03 137210056 IC50 > 10000 nM T40474 CYZ89D 137225046 IC50 > 20000 nM T40474 C1DQG0 137225072 IC50 > 20000 nM T40474 C2TUO4 137283331 IC50 = 0.5 nM T40474 CCS97P 137300718 IC50 = 0.7 nM T40474 CEHT89 137300719 IC50 = 0.7 nM T40474 CXC69T 137321158 IC50 = 92 nM T40474 CE75QD 137321162 IC50 = 15 nM T40474 CCE8N9 137348420 IC50 = 23 nM T40474 C45PIB 137631735 IC50 = 22.39 nM T40474 C25ERN 137631967 IC50 = 196.1 nM T40474 C30ZJV 137632340 IC50 = 9.21 nM T40474 C70BOR 137632456 IC50 = 11.63 nM T40474 CSH8D4 137632523 IC50 = 0.7 nM T40474 CAZW15 137632656 IC50 = 235 nM T40474 C6U2VY 137632775 IC50 = 3.23 nM T40474 CIEQ74 137633008 IC50 = 46.27 nM T40474 CFP02W 137633349 IC50 = 41.23 nM T40474 C2RJM7 137633352 IC50 = 4.3 nM T40474 COC0H4 137633833 IC50 > 10000 nM T40474 CHC70D 137634143 IC50 = 1.06 nM T40474 CI1E8V 137634241 IC50 > 10000 nM T40474 CLG1F2 137634498 IC50 = 0.6 nM T40474 C4CXE7 137635862 IC50 > 10000 nM T40474 CX79FY 137636295 IC50 = 0.5 nM T40474 CD1Y8G 137636528 IC50 = 66.7 nM T40474 CXY4W3 137636605 IC50 = 0.3 nM T40474 C0C6QA 137636845 IC50 = 41.25 nM T40474 C06JRX 137637094 IC50 > 1000 nM T40474 CN0VO5 137637343 IC50 = 33.51 nM T40474 C2WC4O 137637790 IC50 = 12.58 nM T40474 C1FZA0 137639212 IC50 = 0.7 nM T40474 CE96AL 137639657 IC50 > 100000 nM T40474 C5YU7D 137640076 IC50 = 2.6 nM T40474 C37FUH 137640271 IC50 = 0.4 nM T40474 CF13UX 137640338 IC50 = 0.5 nM T40474 C1X5OZ 137641235 IC50 = 35.29 nM T40474 CR6Y5L 137642136 IC50 = 10.46 nM T40474 COF17H 137642341 IC50 > 100 nM T40474 C9HUR8 137642884 IC50 = 455 nM T40474 CKR47C 137643001 IC50 = 278 nM T40474 C9V7NI 137643007 IC50 = 32.15 nM T40474 C6P3OU 137644255 IC50 = 13.14 nM T40474 C67BEV 137644591 IC50 = 18.24 nM T40474 CC31KN 137644869 IC50 = 5.61 nM T40474 CEW37Y 137644947 IC50 = 0.5 nM T40474 C96PQD 137645348 IC50 = 0.7 nM T40474 CVXU72 137645390 IC50 = 8.03 nM T40474 C3YM6A 137645462 IC50 = 237 nM T40474 C13NAH 137645659 IC50 = 46.91 nM T40474 CA4CQ8 137645679 IC50 = 42.15 nM T40474 CT23JE 137645754 IC50 > 100 nM T40474 CN68CK 137647361 IC50 = 39.52 nM T40474 CZ2W1O 137647810 IC50 = 6.76 nM T40474 CNY12B 137648909 IC50 = 10.25 nM T40474 C2L7EN 137649118 IC50 = 1.7 nM T40474 CCP7S5 137649124 IC50 > 10000 nM T40474 C0D9HS 137649160 IC50 = 45.31 nM T40474 C3DMY4 137649270 IC50 = 95 nM T40474 CKU16G 137649619 IC50 = 1078 nM T40474 CH1M9D 137650179 IC50 = 18.26 nM T40474 COAQ87 137650817 IC50 = 258 nM T40474 CDU3P2 137650862 IC50 = 0.9 nM T40474 C1DK0P 137651391 IC50 > 1000 nM T40474 CY1MU9 137651522 IC50 = 14.41 nM T40474 CV9MI4 137652089 IC50 = 0.5 nM T40474 CCQ98L 137652544 IC50 = 29.35 nM T40474 C6YXE3 137652609 IC50 = 18.25 nM T40474 CE6FJ7 137652748 IC50 = 1 nM T40474 CK28XI 137652846 IC50 = 1.5 nM T40474 C3LAD6 137652990 IC50 > 100000 nM T40474 CPQ3I2 137653233 IC50 = 4.52 nM T40474 CU2WN3 137653330 IC50 > 10000 nM T40474 CR0AJ2 137653657 IC50 = 49.16 nM T40474 C05MZI 137655483 IC50 = 2279 nM T40474 CVM9J0 137655717 IC50 = 457 nM T40474 CU8YH3 137655852 IC50 = 5.02 nM T40474 C4G9IS 137655877 IC50 = 1.3 nM T40474 C7U4IK 137656813 IC50 = 8.42 nM T40474 C2JSZ7 137656897 IC50 = 56.25 nM T40474 CC2Q4P 137657659 IC50 = 19.54 nM T40474 C1N2GQ 137657756 IC50 = 2140 nM T40474 CO8W5T 137657796 IC50 = 0.3 nM T40474 CV5H3Z 137657932 IC50 > 1000 nM T40474 CPV1S9 137658287 IC50 = 17 nM T40474 CAHM45 137659715 IC50 = 3.57 nM T40474 C56UJX 137659894 IC50 = 11.23 nM T40474 CBX9G1 137659897 IC50 = 3.8 nM T40474 CN65GR 137660076 IC50 = 19.14 nM T40474 CY3B9N 137660476 IC50 = 3.5 nM T40474 C7KVI0 137660610 IC50 = 36.18 nM T40474 CR1QG6 137660668 IC50 = 2547 nM T40474 CVEF94 137661770 IC50 = 15.27 nM T40474 CZP65E 137661996 IC50 = 0.4 nM T40474 CGX92C 138393291 IC50 = 1100 nM T40474 CSRI06 138547901 IC50 > 1000 nM T40474 CUXO19 138617501 IC50 > 1000 nM T40474 CCT23N 141340950 IC50 = 18 nM T40474 C2ONV6 141370263 EC50 = 11.7 nM T40474 CQ26YL 141370273 EC50 = 2.9 nM T40474 CV9H4O 141370282 EC50 = 32.6 nM T40474 CSF3K7 141370291 EC50 = 1 nM T40474 C6CH2M 141370292 EC50 = 2.3 nM T40474 C0FRL9 141370306 EC50 = 3.8 nM T40474 C7DKV5 141370316 EC50 = 68.3 nM T40474 C43TVS 141370328 EC50 = 3.2 nM T40474 CP1S5N 141370337 EC50 = 3.6 nM T40474 CP0T1D 141370338 EC50 = 2.7 nM T40474 C2WOA3 141370339 EC50 = 1.6 nM T40474 C65GCS 141370343 EC50 = 4.4 nM T40474 CXLN69 141370344 EC50 = 3.4 nM T40474 CU47BN 141370350 EC50 = 4.6 nM T40474 C6C2ZY 141370365 EC50 = 64.5 nM T40474 C8GO0I 141370369 EC50 = 31 nM T40474 CW51PM 141370377 EC50 = 5.9 nM T40474 C7B1JG 141370378 EC50 = 1.7 nM T40474 CD7SI1 141370383 EC50 = 4.5 nM T40474 C90DVN 141391357 IC50 = 1660 nM T40474 C8OTM7 141391358 IC50 = 3900 nM T40474 CJ0A5Q 141391369 IC50 = 2230 nM T40474 COB9P2 141456067 IC50 = 540 nM T40474 CAH02D 141456400 EC50 = 1 nM T40474 C2R3SY 141481761 IC50 = 3.59 nM T40474 CG0S2C 141503867 IC50 = 8.24 nM T40474 C82OQY 141503871 IC50 = 7.06 nM T40474 C53RXW 141503886 IC50 = 12.53 nM T40474 CWB38N 141503895 IC50 = 16.29 nM T40474 CKO04Y 141523342 IC50 = 29.24 nM T40474 CBV02S 141523348 IC50 = 2.86 nM T40474 C73EIP 141523351 IC50 = 31.82 nM T40474 C34CKN 141523354 IC50 = 2.36 nM T40474 CVIM95 141761969 IC50 = 81.7 nM T40474 C98HPQ 141761970 IC50 = 14.5 nM T40474 CY60WS 141761971 IC50 = 154 nM T40474 CJ07NZ 141761972 IC50 = 26.3 nM T40474 C6VB3O 145925651 IC50 >= 5000 nM T40474 C29XUO 145945978 IC50 > 1000 nM T40474 C4HB8M 145949394 IC50 = 21 nM T40474 CB3Z1W 145949428 IC50 = 57.8 nM T40474 C4KZ5S 145949457 IC50 = 15.6 nM T40474 CSR2Z1 145949787 IC50 = 495 nM T40474 CZ3S8A 145950257 IC50 = 13.9 nM T40474 CV92JM 145950565 IC50 = 2350 nM T40474 C2AS8P 145950744 IC50 = 688 nM T40474 CJR79F 145950862 IC50 = 97 nM T40474 CAP0H8 145950928 IC50 = 580 nM T40474 CQ8WP4 145951108 IC50 = 205 nM T40474 CKDS93 145951387 IC50 = 154 nM T40474 C7H9DE 145951575 IC50 = 27030 nM T40474 C0M1IN 145951722 IC50 = 61 nM T40474 CG3SK5 145951952 IC50 = 20690 nM T40474 C36NMP 145952077 IC50 > 50000 nM T40474 CH8K2T 145952204 IC50 = 4100 nM T40474 C15AEX 145952580 IC50 = 358 nM T40474 CM3CX8 145952650 IC50 > 1000 nM T40474 C8V4MP 145952681 IC50 = 731 nM T40474 C8ZQH7 145952959 IC50 = 659 nM T40474 C2P1NK 145953217 IC50 = 348 nM T40474 C3ABQ7 145953222 IC50 = 68 nM T40474 COA5Y3 145953378 IC50 = 820 nM T40474 C65HOU 145953636 IC50 = 37 nM T40474 CJ93IN 145953656 IC50 = 141 nM T40474 CH7I6M 145953803 IC50 = 50 nM T40474 CPY74T 145954284 IC50 = 320 nM T40474 C89RPH 145954372 IC50 = 703 nM T40474 C7ZMS3 145954544 IC50 > 50000 nM T40474 C2N6WX 145954773 IC50 = 415 nM T40474 C74SND 145955336 IC50 = 170 nM T40474 C6JZ7R 145955666 IC50 = 17000 nM T40474 C27KDN 145956212 IC50 = 6510 nM T40474 C5VSC7 145956704 IC50 = 10000 nM T40474 C2V8DA 145957160 IC50 > 1000 nM T40474 CWD5K0 145957408 IC50 = 169 nM T40474 C3CB2R 145957879 IC50 = 196 nM T40474 C42ZQH 145958534 IC50 > 1000 nM T40474 C4C5VP 145958581 IC50 = 809 nM T40474 CXWH23 145958592 IC50 = 967 nM T40474 C7U3TF 145959054 IC50 = 308 nM T40474 CCKZ35 145959119 IC50 = 658 nM T40474 CBQ69R 145959266 IC50 = 94 nM T40474 CE65LI 145959403 IC50 = 1210 nM T40474 CHWG35 145959685 IC50 = 8860 nM T40474 CRYN76 145959686 IC50 = 46 nM T40474 CLSN47 145959907 IC50 = 30 nM T40474 C3ERV5 145959925 IC50 = 5490 nM T40474 C2IHF1 145960158 IC50 = 3350 nM T40474 CV2PA8 145960227 IC50 = 2640 nM T40474 CHYB79 145960278 IC50 = 331 nM T40474 CX35IH 145961002 IC50 = 79.3 nM T40474 CNIE43 145961402 IC50 > 50000 nM T40474 CM46GW 145962083 IC50 = 24000 nM T40474 CJT41L 145962084 IC50 = 73 nM T40474 CI0X7S 145962717 IC50 = 10500 nM T40474 C2CMR3 145963883 IC50 = 59 nM T40474 CRO27A 145964093 IC50 = 5.1 nM T40474 C69JWI 145964256 IC50 > 1000 nM T40474 CIME61 145964672 IC50 = 0.44 nM T40474 C65YWX 145964882 IC50 > 10000 nM T40474 CHC3T0 145965031 IC50 > 10000 nM T40474 CP92ZF 145965329 IC50 = 2100 nM T40474 CPF3U9 145965371 IC50 = 36 nM T40474 COH6A8 145965638 IC50 = 0.54 nM T40474 CMI61S 145965843 IC50 = 52 nM T40474 CZ9QK6 145965864 IC50 = 0.96 nM T40474 CI9R2E 145966320 IC50 = 47 nM T40474 C68UOR 145966334 IC50 = 1.3 nM T40474 C9HXI4 145966620 IC50 > 10000 nM T40474 CQE9M5 145966810 IC50 = 3500 nM T40474 C8O6RY 145966838 IC50 = 1 nM T40474 CN2BE6 145967025 IC50 > 1000 nM T40474 C1EH6C 145967078 IC50 > 10000 nM T40474 CKU36Y 145967168 IC50 > 1000 nM T40474 CYTC61 145967195 IC50 > 1000 nM T40474 CDW83M 145967332 IC50 = 24.4 nM T40474 C0GY3Q 145967784 IC50 = 1.5 nM T40474 CDNC31 145967951 IC50 > 500 nM T40474 C3LH2I 145968221 IC50 = 1 nM T40474 CWJ12M 145969155 IC50 = 420 nM T40474 CGW5S1 145969844 IC50 > 10000 nM T40474 CME7W2 145970049 IC50 = 0.96 nM T40474 CB8R3A 145970271 IC50 > 10000 nM T40474 C18EDZ 145970537 IC50 > 1000 nM T40474 C18ASM 145970764 IC50 = 29.3 nM T40474 CX7DK6 145971283 IC50 = 337 nM T40474 C4EU5J 145971645 IC50 = 37 nM T40474 CD3A7T 145971972 IC50 = 442 nM T40474 C9I5KY 145972522 IC50 > 1000 nM T40474 C9C8SN 145972950 IC50 = 427 nM T40474 C6O7SG 145972970 IC50 = 8.32 nM T40474 C40VIL 145972979 IC50 > 10000 nM T40474 C4GNK0 145973805 IC50 = 114 nM T40474 CQBY19 145974023 IC50 = 6300 nM T40474 CR97YL 145974686 IC50 > 1000 nM T40474 CXRY95 145974888 IC50 = 19 nM T40474 CI2XK9 145975133 IC50 = 2322 nM T40474 CT1XV5 145975325 IC50 > 1000 nM T40474 C74TYP 145975351 IC50 = 2.61 nM T40474 CQXK92 145975423 IC50 = 168.7 nM T40474 CO31CX 145975449 IC50 > 1000 nM T40474 C2NP6U 145975596 IC50 = 0.71 nM T40474 CM7K0A 145975625 IC50 = 25 nM T40474 CXS4L8 145975683 IC50 = 35000 nM T40474 CU48WZ 145976699 IC50 = 136 nM T40474 CICP80 145976788 IC50 > 1000 nM T40474 C8Z2IP 145976817 IC50 = 0.73 nM T40474 C93DAK 145977205 IC50 = 9.89 nM T40474 CSC6A1 145977313 IC50 = 3.7 nM T40474 C4X7CT 145977420 IC50 > 10000 nM T40474 C8DBK1 145977522 IC50 = 1.2 nM T40474 C9LP6T 145977589 IC50 > 1000 nM T40474 CF2D9J 145977619 IC50 = 48 nM T40474 CCD9U2 145977675 IC50 = 0.63 nM T40474 CT92JD 145977767 IC50 > 1000 nM T40474 C9Y1OR 145978262 IC50 = 32 nM T40474 CLA57T 145978300 IC50 > 10000 nM T40474 CR1ZY6 145978627 IC50 = 1.1 nM T40474 C08QWD 145979053 IC50 = 571 nM T40474 CZ0KJ1 145979284 IC50 = 16.83 nM T40474 C6AQ7X 145979475 IC50 = 442 nM T40474 C5TP2U 145979643 IC50 = 907 nM T40474 CDG6Z0 145979655 IC50 > 1000 nM T40474 CP3XF0 145980163 IC50 = 154 nM T40474 CV2QD8 145981005 IC50 = 137 nM T40474 CKQ71E 145981064 IC50 = 2.23 nM T40474 CR39TX 145981127 IC50 = 2.1 nM T40474 CTU32E 145981291 IC50 = 348 nM T40474 CK96JF 145981325 IC50 = 0.71 nM T40474 CS3H2A 145981801 IC50 = 7.97 nM T40474 CE8K2L 145981872 IC50 = 161 nM T40474 CO68TW 145982351 IC50 = 8.53 nM T40474 CFZ06Y 145982656 IC50 = 2.02 nM T40474 CDE94C 145982675 IC50 = 27.3 nM T40474 C87LSD 145982730 IC50 = 16.7 nM T40474 CJK9D7 145983807 IC50 = 150 nM T40474 C8ZVP2 145983956 IC50 > 10000 nM T40474 CTVF58 145984206 IC50 > 10000 nM T40474 C4KJ7X 145984341 IC50 > 10000 nM T40474 C3QYD0 145984532 IC50 > 10000 nM T40474 COC51I 145984537 IC50 = 17.3 nM T40474 CGNE81 145984557 IC50 = 31.4 nM T40474 CN1J7C 145984805 IC50 > 10000 nM T40474 CA8WU3 145984897 IC50 > 1000 nM T40474 CYH09Z 145985311 IC50 = 201 nM T40474 CUM0T5 145985365 IC50 = 14.5 nM T40474 CLGE45 145985395 IC50 = 2.8 nM T40474 C2VJK9 145985408 IC50 > 1000 nM T40474 CEY3K8 145985797 IC50 = 64.9 nM T40474 C35BWZ 145985798 IC50 = 28.6 nM T40474 CR43QN 145985941 IC50 = 110 nM T40474 CHZN24 145986131 IC50 = 440 nM T40474 CGT8I9 145986709 IC50 = 651 nM T40474 CNJ6K9 145986726 IC50 = 38.29 nM T40474 C5KEW2 145986825 IC50 = 678 nM T40474 CHE16J 145986928 IC50 = 364 nM T40474 COD39K 145986975 IC50 = 21.76 nM T40474 C1T9ZV 145987013 IC50 = 241 nM T40474 C1Y5MO 145987062 IC50 = 1.92 nM T40474 CV75AR 145987208 IC50 = 9.2 nM T40474 CM3FP6 145987671 IC50 = 2.7 nM T40474 CRDA10 145987979 IC50 = 456 nM T40474 CNZB43 145987986 IC50 = 32.51 nM T40474 CNG38F 145988243 IC50 = 107.5 nM T40474 CO95CW 145988567 IC50 = 518 nM T40474 C3I8BK 145988938 IC50 > 1000 nM T40474 C81NKP 145989259 IC50 = 836 nM T40474 C4IWH1 145990082 IC50 = 9.25 nM T40474 CQY83A 145990210 IC50 = 177 nM T40474 CJS9Z0 145990229 IC50 = 14 nM T40474 C8PL9Y 145990409 IC50 = 10.05 nM T40474 CI14YQ 145990493 IC50 > 1000 nM T40474 C4YU5L 145990548 IC50 > 1000 nM T40474 CV0N5J 145990633 IC50 = 6.41 nM T40474 CRF53V 145990730 IC50 > 1000 nM T40474 C58ODP 145991046 IC50 = 7.8 nM T40474 C3LB2R 145991081 IC50 = 2.5 nM T40474 CG13QR 145991430 IC50 = 291 nM T40474 CLK61X 145992276 IC50 = 3.8 nM T40474 CY9K6P 145992397 IC50 = 134 nM T40474 CNC69T 145992844 IC50 = 506 nM T40474 C03SEV 145992875 IC50 = 162 nM T40474 COXE84 145992959 IC50 = 550 nM T40474 C14WJN 145993419 IC50 = 260 nM T40474 CG9TY4 145993472 IC50 = 241 nM T40474 CP81CX 146832100 IC50 = 104 nM T40474 CWA71D 149110412 EC50 = 66.59 nM T40474 CS7Q1E 152878273 IC50 = 203 nM T40474 CPV10R 154701379 EC50 = 1.94 nM T40474 CY1ZH2 155510358 IC50 > 10000 nM T40474 C37FPZ 155510738 IC50 > 1500 nM T40474 CEF6A7 155511067 IC50 = 8.1 nM T40474 CD3I9W 155511231 IC50 = 26.71 nM T40474 CQI50K 155511379 IC50 = 94 nM T40474 CL4B2M 155512535 IC50 = 6220 nM T40474 CF0Q2D 155513002 IC50 = 2.1 nM T40474 C81YCJ 155513061 IC50 = 17910 nM T40474 CQA9U6 155513155 IC50 = 18 nM T40474 C2MD1Q 155513187 IC50 > 10000 nM T40474 CZ7K6H 155513660 IC50 = 12000 nM T40474 C8XHM5 155516263 IC50 = 12.6 nM T40474 C2WRO5 155516460 IC50 = 14.7 nM T40474 CTU03S 155516767 IC50 = 0.6 nM T40474 C86HPW 155518524 IC50 = 61000 nM T40474 CJ7KU0 155518881 IC50 = 45.3 nM T40474 CNU28S 155519814 IC50 > 1000 nM T40474 CV2JG7 155520114 EC50 = 18.1 nM T40474 CAR53N 155520426 IC50 = 30.15 nM T40474 C2P0LT 155522675 IC50 > 1000 nM T40474 CK9HR4 155524098 IC50 = 2.56 nM T40474 CG13QJ 155524262 IC50 = 5.5 nM T40474 C5GFE1 155524420 IC50 = 4.7 nM T40474 CPK67I 155524868 IC50 = 2.5 nM T40474 C0COA7 155525819 IC50 = 50 nM T40474 CEV4D0 155526828 IC50 = 21.4 nM T40474 C28YTJ 155527217 IC50 = 2.4 nM T40474 CEQ0F9 155528026 IC50 = 28.1 nM T40474 C8SFQ6 155528028 IC50 = 15 nM T40474 CKBQ85 155528363 IC50 = 132.7 nM T40474 CO3W0R 155528703 IC50 = 2.4 nM T40474 CXDF94 155529218 IC50 = 29.85 nM T40474 CHI54P 155529236 IC50 > 1000 nM T40474 CO28NK 155531294 IC50 = 16 nM T40474 C8CTK0 155532749 IC50 = 2.3 nM T40474 CGVZ73 155532854 IC50 > 1000 nM T40474 C0V9QN 155532882 IC50 = 4500 nM T40474 C6ZE4H 155533175 IC50 = 17.7 nM T40474 C6YQC4 155533269 IC50 = 2.5 nM T40474 C67XEV 155533571 IC50 = 9.8 nM T40474 C7KPE8 155534298 IC50 = 48.54 nM T40474 CM0U3I 155534552 IC50 = 213 nM T40474 CEQJ52 155534874 IC50 = 532 nM T40474 C9FPB6 155535794 IC50 = 140 nM T40474 CE5NI6 155535823 IC50 = 1.42 nM T40474 C2H3PE 155536668 IC50 = 3.9 nM T40474 CZR0J9 155537757 IC50 = 300 nM T40474 CTP72E 155538424 IC50 = 6.3 nM T40474 C1WT0A 155538576 IC50 = 1.7 nM T40474 C9RI7P 155539052 IC50 = 11.8 nM T40474 CAVF74 155539422 IC50 = 63.45 nM T40474 C5WK7Q 155539567 IC50 = 14 nM T40474 C17ORN 155539894 IC50 = 55.39 nM T40474 C14WSM 155540347 EC50 = 91.8 nM T40474 C5N2ST 155541216 IC50 = 25.9 nM T40474 C4LH9J 155541493 IC50 = 29.32 nM T40474 CR59XY 155541644 IC50 = 15.42 nM T40474 CBE29H 155541740 EC50 = 2.79 nM T40474 CBS38V 155541745 EC50 > 1000 nM T40474 C1O0HP 155541936 EC50 = 33.24 nM T40474 C5V0GE 155541941 IC50 = 49.14 nM T40474 C4WKZ0 155542017 EC50 = 17.2 nM T40474 C3HV1C 155542724 EC50 = 7.7 nM T40474 CG6M1N 155543866 EC50 = 37.7 nM T40474 CQ17XT 155543872 IC50 = 24 nM T40474 C2UYB4 155544181 EC50 = 3.3 nM T40474 C5AY1T 155544283 EC50 = 2.5 nM T40474 CR4M1B 155544333 IC50 = 104.9 nM T40474 CT79JF 155545406 IC50 = 4.7 nM T40474 CTW34L 155545445 EC50 = 12.71 nM T40474 C2I6HY 155545590 IC50 = 4.7 nM T40474 C4M2JT 155545755 IC50 = 14.8 nM T40474 C96VGL 155546231 IC50 = 39.64 nM T40474 C9V0RM 155546589 EC50 = 81 nM T40474 CJ6OD0 155546821 EC50 = 15.19 nM T40474 C7SF2C 155547229 IC50 = 1.98 nM T40474 C21SYP 155547261 EC50 = 5.17 nM T40474 CU2VS5 155547607 IC50 = 4.64 nM T40474 C5T6JO 155547777 IC50 = 29.36 nM T40474 CFOY85 155547870 IC50 = 50.26 nM T40474 C60YKA 155548301 IC50 > 1000 nM T40474 C03JOI 155548440 IC50 = 44.78 nM T40474 CLRH45 155549474 EC50 = 10.6 nM T40474 C26AZO 155549906 EC50 = 9.3 nM T40474 CD09XW 155549963 IC50 = 1 nM T40474 CH95WO 155550617 IC50 = 35 nM T40474 CY52AV 155550628 EC50 = 4.9 nM T40474 C9L8DH 155550702 EC50 = 39.2 nM T40474 CI40RU 155550990 IC50 = 9.4 nM T40474 C5IUZ6 155551115 EC50 = 6.41 nM T40474 C5L7HY 155551127 IC50 = 500 nM T40474 CETN42 155552011 IC50 = 4 nM T40474 C1LS4J 155552081 IC50 = 54.24 nM T40474 CN2KX6 155552129 IC50 = 9.87 nM T40474 CS9T5C 155552336 IC50 = 2.34 nM T40474 CZ4J2P 155552610 IC50 = 325 nM T40474 CJ01IF 155553108 IC50 = 54.48 nM T40474 C94JKW 155553894 EC50 = 13.5 nM T40474 CFW6C0 155554557 IC50 = 1.7 nM T40474 CH32NX 155554603 EC50 > 1000 nM T40474 C0BN4R 155556000 IC50 = 34.45 nM T40474 CNOW65 155556826 EC50 = 13.25 nM T40474 C23WLI 155557617 EC50 = 22.5 nM T40474 C10JCL 155557686 EC50 = 2.49 nM T40474 CPZ39X 155558101 EC50 > 1000 nM T40474 CNY35A 155558123 EC50 = 2.74 nM T40474 CO6M9N 155558296 IC50 = 16.07 nM T40474 CDTP67 155558407 EC50 = 3.95 nM T40474 CC8R3X 155558455 IC50 = 65 nM T40474 C9HY2U 155558552 EC50 = 1.6 nM T40474 C7XF4A 155558590 EC50 = 16.4 nM T40474 CCUR26 155559385 EC50 = 9.4 nM T40474 C1OI5K 155559863 IC50 > 1000 nM T40474 CW8BQ2 155559928 EC50 = 38.45 nM T40474 CBA35K 155559950 IC50 = 89 nM T40474 C2CQO9 155560161 EC50 = 11.4 nM T40474 C9E6XB 155560400 EC50 = 28.1 nM T40474 CR3BL5 155561070 IC50 = 5.81 nM T40474 CQ3VN2 155561716 IC50 = 33.8 nM T40474 CC5F3I 155562216 IC50 = 8300 nM T40474 CF3WC6 155562219 IC50 = 1.8 nM T40474 C40IYS 155562258 IC50 = 7.1 nM T40474 CNDL07 155562495 IC50 = 42 nM T40474 CI5UL4 155562624 IC50 = 9.7 nM T40474 CU9AI4 155562673 EC50 = 1.32 nM T40474 CM3P7D 155563249 EC50 = 640.9 nM T40474 CE6IV8 155563850 IC50 = 9.9 nM T40474 COV4D5 155564489 EC50 = 8.7 nM T40474 C2C8VR 155564618 IC50 = 15.6 nM T40474 C5KAN9 155564649 IC50 = 0.7 nM T40474 CTML75 155565088 IC50 = 36.25 nM T40474 C9UNB6 155565959 IC50 = 6.4 nM T40474 CO89GZ 155566463 EC50 = 4.2 nM T40474 C04TDH 155566885 EC50 = 14.1 nM T40474 CT9SY6 155567241 EC50 = 3.67 nM T40474 C01BEA 155567849 EC50 = 100 nM T40474 CI10NL 155567927 IC50 = 25.17 nM T40474 C13LBV 155567954 IC50 = 4.2 nM T40474 C1HKP3 155568631 IC50 = 30.5 nM T40474 CZ9GJ1 155568910 IC50 = 33.2 nM T40474 D00EMH 56597775 IC50 = 26 nM T40474 D00HVA 11624601 Ki > 2900 nM T40474 D00TBD 10461815 IC50 = 9 nM T40474 D02BXJ 46864270 IC50 > 3000 nM T40474 D03DZO 11715767 IC50 > 10000 nM T40474 D03NBX 637308 IC50 = 12900 nM T40474 D03OZD 56671814 Ki = 161 nM T40474 D04CUA 44256277 IC50 = 8 nM T40474 D06HVH 54613583 IC50 > 10000 nM T40474 D06QWO 14824655 IC50 > 10 ug.mL-1 T40474 D07ADX 54764565 IC50 = 177 nM T40474 D07OXC 11650194 IC50 = 8.9 nM T40474 D07SRX 9797919 IC50 > 10000 nM T40474 D08HFG 24809764 IC50 > 10000 nM T40474 D08HGK 3149447 IC50 > 100000 nM T40474 D09HVH 135566652 IC50 > 10 nM T40474 D09RYV 9911652 IC50 > 20000000 nM T40474 D09TNR 9850161 IC50 > 10000 nM T40474 D0A1CM 5281855 IC50 = 580 nM T40474 D0E1QI 9549297 IC50 = 10 nM T40474 D0G3SZ 6918469 IC50 = 4.3 ug.mL-1 T40474 D0J3LR 11634725 Ki > 4000 nM T40474 D0K4ZR 11652416 IC50 = 5500 nM T40474 D0L3JR 25212148 IC50 = 20 nM T40474 D0M4SY 135440466 IC50 = 4870 nM T40474 D0ME9B 46868971 IC50 > 10 nM T40474 D0N5XG 45267314 IC50 = 19 nM T40474 D0OZ2S 11785878 IC50 > 10000 nM T40474 D0Q3NG 11715520 Ki > 2900 nM T40474 D0R2WK 16038120 IC50 = 1667 nM T40474 D0RO9R 50942314 IC50 = 44 nM T40474 D0S0GT 22028181 IC50 = 1175 nM T40474 D0S1II 45272467 IC50 = 250 nM T40474 D0S7IE 11658882 Ki > 2900 nM T40474 D0T8NU 16757525 IC50 > 4000 nM T40474 D0U4JW 45270766 IC50 = 3500 nM T00420 CAT8Q3 3000500 IC50 = 6000 nM T00420 CV7Q9E 155511454 IC50 > 100000 nM T00420 CI0SQ9 155516407 IC50 = 1000 nM T00420 CB4PM0 155527954 IC50 = 32000 nM T00420 CV24FT 155528313 IC50 = 25000 nM T00420 CRO73G 155531931 IC50 = 25000 nM T00420 C4YW6O 155540732 IC50 = 19000 nM T00420 C9RBY6 155540926 IC50 = 31000 nM T00420 CQ61HG 155546548 IC50 = 70000 nM T00420 C85ABG 155549837 IC50 = 63000 nM T00420 C4L5NQ 155558307 IC50 = 17000 nM T00420 CG5V2Z 155561482 IC50 > 100000 nM T00420 C8Y9QV 155561966 IC50 = 19000 nM T00420 C9V1QH 155562398 IC50 > 100000 nM T00420 D0I1NU 72392 IC50 = 21000 nM T15514 CW65TR 50354 EC50 = 2090 nM T15514 CL3Q7C 53424 EC50 = 2570 nM T15514 CAYT42 53425 EC50 = 2330 nM T15514 CV4UA6 55507 EC50 = 1950 nM T15514 C5RWK7 55508 EC50 = 1280 nM T15514 CC3Z1N 56909 EC50 = 1220 nM T15514 CI6M7O 100603 EC50 = 1470 nM T15514 CT8B3W 2990364 EC50 > 100000 nM T17228 D01SHZ 9931954 IC50 = 407.38 nM T17228 D0J9HW 23725625 IC50 = 46 nM T17228 D00BMF 24958200 IC50 = 295.12 nM T17228 CXG7Y0 76959 IC50 > 100000 nM T17228 CJ2UB5 236501 IC50 > 100000 nM T17228 CR26SK 4163640 IC50 = 50000 nM T17228 CT9V6M 4826644 IC50 = 34000 nM T17228 C4P2UQ 8607850 IC50 > 100000 nM T17228 CI0QP9 11960529 IC50 = 2137.96 nM T17228 C1Y2MX 24772013 IC50 = 70 nM T17228 CL8Q0K 24772834 IC50 = 50 nM T17228 C0IOR9 25015515 IC50 = 1288.25 nM T17228 CMXA39 28825277 IC50 = 86000 nM T17228 CSO1Z6 28825295 IC50 > 100000 nM T17228 C7QLY3 71464718 IC50 > 10000 nM T17228 C24XZF 71576800 IC50 > 10000 nM T17228 C3XO5D 89649815 IC50 > 100000 nM T17228 C2XR5Q 92045137 IC50 = 46 nM T17228 CV0NZ7 105539834 IC50 > 100000 nM T17228 C02SDC 122423373 IC50 = 2800 nM T17228 CV06MU 131801402 IC50 > 100000 nM T17228 C47LAF 135418940 IC50 = 831.76 nM T17228 CQ06WL 135566761 IC50 = 1300 nM T17228 CT8NG2 135566762 IC50 > 100000 nM T17228 C1L2WD 135566841 IC50 = 2200 nM T17228 C8PQM0 135566842 IC50 = 1000 nM T17228 C7N1YX 135566845 IC50 = 9600 nM T17228 C08WVI 135566846 IC50 = 2200 nM T17228 CU2I7X 135567125 IC50 = 39810.72 nM T17228 C37PTU 135567126 IC50 = 45000 nM T17228 COYA14 135670654 IC50 = 13200 nM T17228 CIL7K3 135742498 IC50 = 62.8 nM T17228 CPW1F0 135893474 IC50 = 14400 nM T17228 C19ZFB 135901558 IC50 > 100000 nM T17228 C4ODX8 135901559 IC50 > 100000 nM T17228 CW7JB0 136229577 IC50 = 15200 nM T17228 C18MSY 136236981 IC50 = 1900 nM T17228 C79TCS 136249352 IC50 = 3800 nM T17228 C35VUY 136264437 IC50 = 11100 nM T17228 CX7PZ5 141639950 IC50 > 100000 nM T17228 D04QRM 135566764 IC50 = 900 nM T17228 D04WDX 4858 IC50 = 1445.44 nM T42337 D08QCJ 5430 EC50 = 3400 nM T42337 D0KG9M 19910 IC50 > 15000 nM T42337 D06WEB 9892113 IC50 = 700 nM T42337 CB4Z9P 1474 EC50 = 320 nM T42337 CH93VI 2817 IC50 = 12900 nM T42337 C1KG9Z 6792 IC50 > 15000 nM T42337 CSU40C 6855 IC50 = 42800 nM T42337 CS0TL4 13224 IC50 > 15000 nM T42337 CF95CG 39492 Ki = 2000 nM T42337 CX43ZG 74464 Ki = 10000 nM T42337 CYZ8T1 93617 Ki > 100000 nM T42337 C7MQ9Z 98449 Ki = 111600 nM T42337 CB7X1C 100489 IC50 = 28800 nM T42337 CFO0Z8 161167 IC50 = 44900 nM T42337 C8YO4C 204802 IC50 = 23400 nM T42337 C1N8YT 241129 Ki = 162000 nM T42337 CUF24Q 262410 Ki = 2000 nM T42337 C9FU7M 319883 Ki > 100000 nM T42337 C8QL7M 319887 Ki > 100000 nM T42337 C5HCU4 338261 Ki = 8000 nM T42337 CDSV18 367144 Ki = 2000 nM T42337 CVH18S 421108 IC50 > 50000 nM T42337 COPG12 448288 IC50 = 14000 nM T42337 C2L7DI 453059 EC50 = 410 nM T42337 CUQ70N 453063 EC50 = 870 nM T42337 C7OB8F 461360 IC50 = 41200 nM T42337 CB5A1S 612049 IC50 = 32400 nM T42337 C2GEC7 661949 EC50 = 49 nM T42337 CL9Q6A 676832 Ki = 6000 nM T42337 CY46ZP 676834 Ki > 100000 nM T42337 CEN1Q2 677067 Ki > 100000 nM T42337 C6O0MF 678009 Ki > 100000 nM T42337 C4TNA0 683337 IC50 > 50000 nM T42337 C62CVW 699784 IC50 > 50000 nM T42337 C32LWZ 708284 Ki > 100000 nM T42337 C7NFI8 727420 Ki = 9000 nM T42337 C7CJF8 727442 Ki = 98000 nM T42337 CNXW91 727443 Ki > 100000 nM T42337 C8WJB4 732234 Ki > 100000 nM T42337 C2KA1Z 843608 Ki > 100000 nM T42337 CULO53 930716 EC50 = 1500 nM T42337 CY4N9Q 935986 EC50 = 110 nM T42337 C8HIA7 937982 EC50 = 940 nM T42337 CWNG75 1070711 IC50 = 8100 nM T42337 C0YG5N 2179724 Ki > 100000 nM T42337 CZX98P 2241752 Ki > 100000 nM T42337 CDU91J 2319832 Ki > 100000 nM T42337 C3AI7O 2725962 IC50 = 1000 nM T42337 CU61SY 2725966 EC50 = 280 nM T42337 C8Q6VT 2725991 IC50 > 100000 nM T42337 CTS7L9 2725999 IC50 = 11000 nM T42337 CS02AC 2740170 IC50 = 8900 nM T42337 C15MSF 2740173 IC50 = 1500 nM T42337 C6OE0C 2740174 EC50 = 190 nM T42337 C79RPV 2784955 Ki > 100000 nM T42337 CAHV18 2795593 IC50 = 1100 nM T42337 C9NOS2 2796249 IC50 = 360 nM T42337 CGI28F 2818423 EC50 = 390 nM T42337 CE49YH 3097900 Ki = 5000 nM T42337 C1UJE2 4068684 IC50 > 15000 nM T42337 CQ2RS5 5292673 Ki = 10000 nM T42337 CCMR86 5326770 IC50 = 370 nM T42337 C6MD2A 5338637 Ki > 100000 nM T42337 CH3NE4 5358573 Ki > 100000 nM T42337 C4SGX7 5879692 Ki = 10 nM T42337 C49OGD 6111416 Ki = 1000 nM T42337 CZOJ84 6612277 IC50 = 27600 nM T42337 CL81SX 9922371 IC50 = 84000 nM T42337 CO52UI 10006629 IC50 > 10000 nM T42337 C3MEL0 10013353 IC50 = 16000 nM T42337 C3J6BM 10059183 IC50 = 19000 nM T42337 C95BKD 10077016 IC50 = 700 nM T42337 CXEO87 10103872 IC50 = 7000 nM T42337 CMC03E 10425401 Ki = 33000 nM T42337 CFI63J 10650951 IC50 = 3000 nM T42337 CGDI42 10797325 IC50 = 18800 nM T42337 C8KCV1 10911160 IC50 = 3500 nM T42337 C6CJ9X 11126767 IC50 = 30100 nM T42337 C7IDU1 11513930 IC50 = 40100 nM T42337 C0X6YF 11535861 IC50 = 35500 nM T42337 CBZ89Y 11543088 IC50 = 37300 nM T42337 CO5H8S 11557818 IC50 = 48500 nM T42337 CNV16Y 11564819 IC50 = 32600 nM T42337 C1P9QY 11587570 IC50 = 41000 nM T42337 C7D4JU 11601120 IC50 = 47000 nM T42337 CXI7A0 11629844 Ki = 4900 nM T42337 CM9ZF4 11629922 Ki = 9900 nM T42337 C5XJQ8 11629988 IC50 = 38800 nM T42337 C42QWY 11644224 IC50 = 45800 nM T42337 C9FZK3 11680001 IC50 = 33900 nM T42337 C9OZA1 11715385 IC50 = 19000 nM T42337 CN9D1L 11809364 EC50 = 350 nM T42337 C53AIB 14744934 Ki > 100000 nM T42337 C30OLU 15083575 Ki > 500000 nM T42337 CBUC49 15516886 IC50 = 63000 nM T42337 CDC80H 15516888 IC50 = 100000 nM T42337 C4DV3T 20660272 IC50 = 69000 nM T42337 C4YUS0 23647754 IC50 = 2200 nM T42337 CH89QX 23647755 IC50 = 12000 nM T42337 CD6Q5V 23647756 IC50 = 8700 nM T42337 CCN67D 23647757 IC50 = 8100 nM T42337 C2P9OQ 44378659 Ki = 390000 nM T42337 CLRN70 44378660 Ki = 48000 nM T42337 C9DC4A 44378725 Ki = 180000 nM T42337 CRD8O0 44381636 IC50 = 12000 nM T42337 CZ6RG7 44381638 IC50 = 46000 nM T42337 CSQ0W5 44381639 IC50 = 89000 nM T42337 C70VGJ 44381640 IC50 = 101000 nM T42337 CR7J1I 44381648 IC50 = 5300 nM T42337 CXW14E 44381649 IC50 = 90000 nM T42337 CA27TF 44381668 IC50 = 34000 nM T42337 CNJ74O 44381669 IC50 = 11000 nM T42337 C1UIR6 44381689 IC50 = 137000 nM T42337 CE82LP 44381690 IC50 > 100000 nM T42337 C0S9NU 44381720 IC50 = 12000 nM T42337 C0TI6L 44381731 IC50 = 66000 nM T42337 C46EFV 44381733 IC50 = 13000 nM T42337 CLA25E 44381734 IC50 = 14000 nM T42337 CX7KI3 44381742 IC50 = 81000 nM T42337 CL0KD5 44381743 IC50 = 4700 nM T42337 CC1PK9 44381755 IC50 = 11000 nM T42337 C4PTD7 44381756 IC50 = 69000 nM T42337 C5GTW7 44381764 IC50 = 63000 nM T42337 C4SNP1 44381771 IC50 = 6800 nM T42337 C9YH2Q 44381772 IC50 = 53000 nM T42337 C1XCO0 44381773 IC50 = 11000 nM T42337 CO60XF 44381796 IC50 > 100000 nM T42337 C9WBI4 44381812 IC50 = 20000 nM T42337 CPQK86 44381823 IC50 = 57000 nM T42337 CZR3U0 44381824 IC50 > 100000 nM T42337 CKS79L 44381893 IC50 > 100000 nM T42337 C5APZ6 44381897 IC50 = 32000 nM T42337 C1BCZ9 44381901 IC50 > 100000 nM T42337 CUP5A0 44381903 IC50 > 100000 nM T42337 CW3I2S 44381904 IC50 = 45000 nM T42337 CA2F3C 44381909 IC50 = 1600 nM T42337 CNMH89 44381916 IC50 = 84000 nM T42337 CSB3V8 44381933 IC50 = 19000 nM T42337 CQR38H 44381935 IC50 = 24000 nM T42337 CAXC40 44381941 IC50 = 75000 nM T42337 CNE58C 44381946 IC50 = 1500 nM T42337 C91HWB 44381954 IC50 = 93000 nM T42337 C63FRA 44381955 IC50 > 100000 nM T42337 CT5GL2 44381961 IC50 = 8900 nM T42337 CK7N0V 44381963 IC50 = 1700 nM T42337 C12GXS 44381973 IC50 = 15000 nM T42337 CC9I0D 44381976 IC50 = 12000 nM T42337 C8JEP3 44381987 IC50 = 12000 nM T42337 C7MHO1 44381988 IC50 = 63000 nM T42337 CZX82N 44381997 IC50 = 1300 nM T42337 CO18AS 44381998 IC50 = 1300 nM T42337 CDX0N9 44381999 IC50 = 5000 nM T42337 C9NE3W 44382027 IC50 = 58000 nM T42337 CGS36C 44382028 IC50 = 68000 nM T42337 CJR46W 44382074 IC50 = 76000 nM T42337 C7WK8D 44382075 IC50 > 100000 nM T42337 CR3TX2 44382078 IC50 = 95000 nM T42337 CNMF84 44382132 IC50 = 18000 nM T42337 CD63HL 44382395 IC50 = 16000 nM T42337 C7HA9B 44382396 IC50 = 78000 nM T42337 C6ZPD8 44382483 IC50 = 13000 nM T42337 C0OZ1L 44382517 IC50 > 100000 nM T42337 C1UE5V 44382789 IC50 = 79000 nM T42337 C83QND 44590979 IC50 > 100000 nM T42337 CU32GN 45267083 IC50 = 3000 nM T42337 CD8MS7 49797979 IC50 = 39800 nM T42337 C9ET7S 51035427 IC50 = 3590 nM T42337 CD9M2G 51035429 IC50 = 5580 nM T42337 C61BNS 53326951 Ki = 54800 nM T42337 C2U0HQ 54602731 IC50 = 27000 nM T42337 CX4A7W 56563890 IC50 > 100000 nM T42337 C4HO0Y 58198133 IC50 = 12200 nM T42337 COU9T2 58279815 IC50 = 100 nM T42337 CB31IC 58279829 IC50 = 10000 nM T42337 C2M9SU 68347001 EC50 = 1600 nM T42337 CI1J8B 68347004 EC50 = 7600 nM T42337 C7VK9T 68347007 IC50 = 600 nM T42337 C6S0MJ 68347012 IC50 = 800 nM T42337 CR60HY 68347026 IC50 = 1100 nM T42337 CF7A0K 68347055 IC50 = 1300 nM T42337 C4I5BQ 68347057 EC50 = 330 nM T42337 CFKS17 68347135 IC50 = 800 nM T42337 C7HS6V 68347136 IC50 = 4600 nM T42337 CT5W9F 68347138 IC50 = 1400 nM T42337 COS5C6 68347139 IC50 = 800 nM T42337 CZRK60 68347140 IC50 = 600 nM T42337 CT19PO 68347143 IC50 = 1700 nM T42337 C2Y0IB 68347313 IC50 = 1100 nM T42337 C26ZEC 68347339 EC50 = 730 nM T42337 CBW2J3 71457398 IC50 = 7450 nM T42337 CI05VW 71459255 IC50 = 5140 nM T42337 CL8H2B 71602394 EC50 = 530 nM T42337 C5TPO1 71602459 EC50 = 1700 nM T42337 C5LCD8 71602460 EC50 = 700 nM T42337 CCB58N 71602527 EC50 = 160 nM T42337 CMWJ83 71602528 EC50 = 1300 nM T42337 CKBD52 71602529 EC50 = 670 nM T42337 CDKF42 71602530 EC50 = 220 nM T42337 C31MVT 71602531 EC50 = 260 nM T42337 CC78SK 71602588 EC50 = 93 nM T42337 C7CT2W 71602589 EC50 = 260 nM T42337 C61ABC 71602590 EC50 = 200 nM T42337 CXCQ63 71602591 EC50 = 780 nM T42337 CBN17L 71602592 EC50 = 710 nM T42337 C7WA2F 71602646 EC50 = 570 nM T42337 CVG89D 71602647 EC50 = 520 nM T42337 CC2R3T 71602648 EC50 = 1200 nM T42337 CP60LJ 71602649 EC50 = 330 nM T42337 C5UP7K 71602650 EC50 = 380 nM T42337 C1UV4S 71602693 EC50 = 420 nM T42337 CGTV32 71602694 EC50 = 690 nM T42337 CV5XT2 71602695 EC50 = 500 nM T42337 CY5S8M 71602696 EC50 = 63 nM T42337 C5ZGU1 71602697 EC50 = 160 nM T42337 C0WOA4 71602745 EC50 = 2300 nM T42337 CM2VE7 71602796 EC50 = 200 nM T42337 CQ6Y1W 71603176 EC50 = 20000 nM T42337 CY60QJ 71603177 EC50 = 7200 nM T42337 COE76Q 71603178 EC50 = 2500 nM T42337 CZM7C8 71603179 EC50 = 270 nM T42337 C20ZQI 71603235 EC50 = 49 nM T42337 CSF38G 71603236 EC50 = 36 nM T42337 CLXH32 71603237 EC50 = 300 nM T42337 CV5Q1A 71603238 EC50 = 140 nM T42337 CE0GO2 71815258 IC50 > 10000 nM T42337 CCF61D 71815827 IC50 > 10000 nM T42337 CSLT73 71815970 IC50 > 10000 nM T42337 CE8A4J 71816100 IC50 > 10000 nM T42337 C1T8FH 73189806 Ki > 500000 nM T42337 CLG1E3 73345794 EC50 = 900 nM T42337 C2WP7O 73345795 EC50 = 6000 nM T42337 CNKZ64 73345796 EC50 = 94 nM T42337 CCUG98 73345797 EC50 = 81 nM T42337 C0C8JI 73345798 EC50 = 590 nM T42337 C9DLK6 73345799 EC50 = 430 nM T42337 C64ZSF 73347280 EC50 = 94 nM T42337 CN90YL 73347281 EC50 = 110 nM T42337 C1EV2G 73347282 EC50 = 1400 nM T42337 CH0IL4 73348796 EC50 = 250 nM T42337 CUH1J4 73348797 EC50 = 93 nM T42337 CU20ZW 73350374 EC50 = 73 nM T42337 CG2K3V 73351884 EC50 = 850 nM T42337 C4N9JC 73353354 EC50 = 120 nM T42337 CT41OK 73353355 EC50 = 120 nM T42337 CAK6B5 73353356 EC50 = 100 nM T42337 C5B3JW 73356423 EC50 = 390 nM T42337 CN58LK 73356424 EC50 = 180 nM T42337 CS3WJ6 85804502 IC50 = 19700 nM T42337 COT8P7 89855771 IC50 > 10000 nM T42337 C7HP6U 89855775 IC50 > 10000 nM T42337 CY7DH8 89855776 IC50 > 10000 nM T42337 CJN31S 89855779 IC50 > 10000 nM T42337 C84GQR 89855793 IC50 > 10000 nM T42337 CC2EV5 89855828 IC50 > 10000 nM T42337 CJ7G3L 89855860 IC50 > 10000 nM T42337 C17GAX 89855873 IC50 > 10000 nM T42337 C32LKW 89855916 IC50 > 10000 nM T42337 CQ63GB 89855918 IC50 > 10000 nM T42337 C72SHX 89855938 IC50 > 10000 nM T42337 CK67TU 89855943 IC50 > 10000 nM T42337 CGU58D 89855953 IC50 > 10000 nM T42337 C7F2UR 89893622 IC50 > 10000 nM T42337 CCN1E5 89893636 IC50 > 10000 nM T42337 CE3NI5 89893683 IC50 > 10000 nM T42337 C6GOP2 89893744 IC50 > 10000 nM T42337 CP37LV 117832568 IC50 > 10000 nM T42337 CE0N7J 118714883 IC50 = 48000 nM T42337 CJZ4Y9 118714885 IC50 = 43000 nM T42337 C0AHF4 118714887 IC50 = 16200 nM T42337 CZS4P5 118714889 IC50 = 12900 nM T42337 CM24NS 118714891 IC50 = 3500 nM T42337 CUM18D 118714893 IC50 = 53700 nM T42337 CQCX50 118714894 IC50 = 16500 nM T42337 CJ97GO 118714897 IC50 = 1000 nM T42337 CE3PN1 118870023 IC50 > 10000 nM T42337 CVD8B4 118884324 IC50 > 10000 nM T42337 CXP15S 130307835 IC50 > 10000 nM T42337 CNGV45 130307851 IC50 > 10000 nM T42337 D02ADV 594397 IC50 = 7100 nM T42337 D02APY 448285 IC50 = 56000 nM T42337 D04MIY 186763 IC50 = 48800 nM T42337 D05DCQ 9838682 Ki = 3900 nM T42337 D07PXR 11665659 IC50 = 34700 nM T42337 D08AXA 947740 IC50 = 10300 nM T42337 D0C0UB 345772 IC50 = 32600 nM T42337 D0FO2B 1923 IC50 = 12900 nM T42337 D0I6RL 11723962 IC50 = 47000 nM T42337 D0L4YF 70821 IC50 = 28400 nM T65755 D00SQN 12136798 IC50 = 7160 nM T65755 D03RTS 2662 IC50 = 1637 nM T65755 D06XGW 12035 IC50 = 3160000 nM T65755 D07POC 176870 IC50 > 15800 nM T65755 D08CDI 208908 IC50 > 100000 nM T65755 D09LNI 3365 IC50 > 40000 nM T65755 D0AZ3C 5291 EC50 > 100000 nM T65755 D0E3SH 6918837 IC50 = 0.83 nM T65755 D0E7PQ 5311 IC50 = 11.5 nM T65755 D0G6QF 3081361 IC50 > 10000 nM T65755 D0L7LC 5352062 IC50 = 15 nM T65755 D0P2GK 5258 Ki = 6340 nM T65755 D0Y3KG 3121 Ki = 564000 nM T65755 D05HWN 16736529 IC50 > 1000 nM T65755 D06TKI 49857317 Ki = 4.8 nM T65755 D07KDI 6918848 IC50 = 16 nM T65755 D07SDQ 969516 IC50 = 187000 nM T65755 D0B3FV 6445533 IC50 = 32 nM T65755 D0B7CH 4775 Ki = 2800 nM T65755 D0C9XA 119 Ki = 8190 nM T65755 D0E3LP 5113032 IC50 > 100000 nM T65755 D0E6UZ 54575456 IC50 = 6.8 nM T65755 D0I7IB 5222465 IC50 = 140000 nM T65755 D0L2UQ 49855250 IC50 = 126 nM T65755 D0M8FD 4261 IC50 = 233 nM T65755 D0XT6W 6918638 IC50 = 26.4 nM T65755 D0Z4RC 24756910 IC50 = 4.4 nM T65755 D0DO5U 9799221 IC50 = 205 nM T65755 D0J8OC 5186 IC50 = 560 nM T65755 D0UL5X 6918714 IC50 = 172 nM T65755 D00OWF 5280953 IC50 > 10000 nM T65755 D0JY1I 42613483 EC50 = 4200 nM T65755 D0V5IQ 130227480 IC50 = 36 nM T65755 D0N3SH 4996 IC50 = 200 nM T65755 D0W9NH 2746 EC50 = 3810 nM T65755 CIJE65 3810 IC50 > 10000 nM T65755 C6FBI7 3811 IC50 = 110 nM T65755 CYEP10 3812 IC50 = 2180 nM T65755 C8HA6K 3994 IC50 = 46 nM T65755 C6XBJ2 4871 IC50 = 1050 nM T65755 CN1YZ9 5044 IC50 > 10000 nM T65755 C5S2BK 5048 EC50 = 1000 nM T65755 C7LH1Z 95168 IC50 = 6530 nM T65755 CLY6K3 661302 IC50 > 100000 nM T65755 CBC31X 817096 IC50 = 51286.14 nM T65755 C96GFC 1798422 IC50 = 12600 nM T65755 C1YQT9 2798084 IC50 = 251.19 nM T65755 CR1Z4O 2798087 IC50 = 125.89 nM T65755 CJ0T4E 3612016 IC50 > 100000 nM T65755 C98ICJ 4157424 IC50 = 102000 nM T65755 C29CSA 4871646 IC50 = 515 nM T65755 CR5Y8E 5226635 IC50 > 10000 nM T65755 C5N4CF 5278571 IC50 = 3800 nM T65755 CDIN74 5278572 IC50 = 3900 nM T65755 CJZW25 5278573 IC50 = 2400 nM T65755 CL5J4B 5278574 IC50 = 3800 nM T65755 C81FUM 5280633 IC50 = 170400 nM T65755 CN4M6D 5281220 IC50 = 18500 nM T65755 C7KAR5 5353765 IC50 = 30 nM T65755 CH5FO1 5353767 IC50 = 59 nM T65755 CSIJ53 5793932 IC50 = 8200 nM T65755 CSA24L 6474310 IC50 = 143240 nM T65755 CXA1J9 6678454 EC50 = 34000 nM T65755 CVH27G 6918801 IC50 = 30 nM T65755 C1RD7E 6918878 IC50 = 204 nM T65755 CE9LP2 9543539 IC50 = 78000 nM T65755 CO3PE1 9543540 IC50 = 87000 nM T65755 CKZ04O 9543541 IC50 = 238000 nM T65755 CY71SA 9543542 IC50 = 204000 nM T65755 CD2AE5 9543543 IC50 = 500000 nM T65755 CUJ32X 9543544 IC50 = 186000 nM T65755 CQR09K 9543545 IC50 = 123000 nM T65755 CE6QY8 9543546 IC50 = 99000 nM T65755 C03CWX 9543547 IC50 = 140000 nM T65755 CO3ZC8 9543548 IC50 = 470000 nM T65755 C7E5KO 9543549 IC50 = 54000 nM T65755 CN8YD7 9543550 IC50 = 438000 nM T65755 C7CFP3 9543551 IC50 = 17000 nM T65755 C0FE9D 9543552 IC50 = 84000 nM T65755 C5OF7J 9543553 IC50 = 91000 nM T65755 CEX68U 9543554 IC50 > 1000 nM T65755 C18VOF 9543555 IC50 = 387000 nM T65755 CDQA28 9543556 IC50 = 14000 nM T65755 C58GIH 9797137 IC50 = 44 nM T65755 CTDA68 9797425 IC50 = 3450000 nM T65755 CJ07ZA 9800555 IC50 = 900 nM T65755 CQU47Z 9814479 IC50 = 22850 nM T65755 CVQ72P 9815480 IC50 = 279 nM T65755 CU43MV 9816273 IC50 = 28 nM T65755 CA9I8J 9817551 IC50 = 28 nM T65755 CV3H9Q 9821324 IC50 = 8 nM T65755 CUP46A 9822443 IC50 = 9.1 nM T65755 CAKY97 9823037 IC50 = 30 nM T65755 C25PSA 9835852 IC50 = 16595.87 nM T65755 CBV96W 9836655 IC50 = 29 nM T65755 CP61TN 9841246 IC50 = 10 nM T65755 CLYJ85 9848223 IC50 = 750 nM T65755 CCU5K3 9857639 IC50 = 625 nM T65755 CL9G7V 9858973 IC50 = 20 nM T65755 C8G6AI 9858986 IC50 = 16 nM T65755 C59GXB 9862144 IC50 = 265 nM T65755 C6OT8D 9870729 IC50 = 38 nM T65755 C45ZYB 9879458 IC50 = 29 nM T65755 CK17CR 9880674 IC50 = 18 nM T65755 CPS24V 9880847 IC50 = 63 nM T65755 CITY43 9882059 IC50 = 20 nM T65755 C0MG5Q 9887245 EC50 = 10000 nM T65755 CSW4Y1 9891541 IC50 = 970 nM T65755 C3T6WU 9901621 IC50 = 29 nM T65755 CS4L7Z 9902895 IC50 = 13 nM T65755 CXIC76 9903149 IC50 = 201 nM T65755 C81EYJ 9923508 IC50 = 8 nM T65755 CQG4V8 9924543 IC50 = 5 nM T65755 CQET03 9945208 IC50 = 7 nM T65755 CCG98N 9952732 IC50 = 6.8 nM T65755 CVK2I0 9967396 IC50 = 34 nM T65755 CVH05G 9969900 IC50 = 23 nM T65755 COE6R7 9972242 IC50 = 14.6 nM T65755 CAV43O 9977314 IC50 = 310 nM T65755 CTYI59 9977701 IC50 = 2800 nM T65755 C4J6YE 9977875 IC50 = 7 nM T65755 C9V4EM 9993471 IC50 = 260 nM T65755 CNB31H 9994119 IC50 = 1200 nM T65755 C3ZQ9T 10001038 IC50 = 8 nM T65755 CMDU83 10002709 IC50 = 9400 nM T65755 CZK3B7 10023483 IC50 = 300 nM T65755 CWH4U2 10055830 IC50 = 27000 nM T65755 CQ8GL7 10062255 IC50 = 5400 nM T65755 CYV8Z0 10063584 IC50 = 380 nM T65755 CN3C0L 10070262 IC50 = 12 nM T65755 CHGX49 10075681 IC50 = 4990 nM T65755 C0R1GC 10081950 IC50 = 22 nM T65755 CX81ML 10092736 IC50 = 4600 nM T65755 C7LP1F 10093090 IC50 = 12 nM T65755 CM9UQ1 10109962 EC50 = 25000 nM T65755 CT2Q0B 10125717 IC50 = 830 nM T65755 C1OPT9 10126993 IC50 = 22 nM T65755 C4ID5Y 10127077 IC50 = 187 nM T65755 C90TQC 10131653 IC50 = 476 nM T65755 CJ2U1E 10134605 IC50 = 10 nM T65755 CWA9R2 10135838 IC50 = 1995 nM T65755 C6ZOI4 10151472 IC50 = 269 nM T65755 CL4C9H 10154438 IC50 = 233.15 nM T65755 CS7EV8 10157466 IC50 = 54 nM T65755 CR1G8D 10157889 EC50 = 5000 nM T65755 CMJ98G 10172225 IC50 = 240 nM T65755 C0M6RD 10172825 IC50 = 84 nM T65755 CN8S3K 10193364 IC50 = 2000 nM T65755 CC5WG3 10193406 IC50 = 9549.93 nM T65755 CUX59I 10194570 IC50 = 212 nM T65755 CPF4J3 10194639 IC50 = 149 nM T65755 CHFY72 10209646 IC50 = 17 nM T65755 C3C7PR 10215484 IC50 = 310 nM T65755 C92QBP 10237760 IC50 = 191 nM T65755 C8WGZ7 10241991 IC50 = 48 nM T65755 CMSX84 10246177 IC50 = 123 nM T65755 CHWT92 10246670 IC50 = 14000 nM T65755 CON61Q 10246764 IC50 = 21 nM T65755 CY2CR9 10246779 IC50 = 33 nM T65755 C5ZAP8 10249964 IC50 = 49 nM T65755 CYX8H4 10266202 IC50 = 150 nM T65755 CY9M6O 10267576 IC50 = 2400 nM T65755 C6B0LJ 10269218 IC50 = 22 nM T65755 C82BPN 10269384 EC50 = 5000 nM T65755 C0LQC5 10269458 IC50 = 42 nM T65755 CK3I9Y 10271952 IC50 = 66 nM T65755 CR07KF 10286983 IC50 = 1.5 nM T65755 C09JQO 10287354 IC50 = 123 nM T65755 CE1UJ8 10309124 IC50 = 1100 nM T65755 CU63CM 10309493 IC50 = 132 nM T65755 C7RC1E 10309899 IC50 = 6 nM T65755 C9L3PX 10310040 IC50 = 68 nM T65755 CP5D1Y 10341900 EC50 = 5000 nM T65755 CJ2T6U 10357349 IC50 = 180 nM T65755 C4DZ3X 10378404 IC50 = 1600 nM T65755 CLM3Z9 10379137 IC50 = 100 nM T65755 C8TS0V 10380251 IC50 = 12187 nM T65755 CJFM96 10401611 IC50 = 1900 nM T65755 CH75UT 10402906 IC50 = 5300 nM T65755 C38YIE 10403253 IC50 = 3440000 nM T65755 C94UQJ 10412869 IC50 = 2 nM T65755 CO9L2E 10426019 IC50 = 2.1 nM T65755 C4MZY2 10429614 IC50 = 60 nM T65755 C6Z5PO 10458209 IC50 = 400 nM T65755 CY9I0S 10470023 IC50 = 153 nM T65755 CW2X8Z 10474722 IC50 = 2200 nM T65755 CPI87X 10479996 IC50 = 51 nM T65755 CX60YL 10502119 IC50 > 100000 nM T65755 C2LJC1 10531767 IC50 = 0.005 ug.mL-1 T65755 CX2KA5 10572471 IC50 > 100000 nM T65755 CPC50T 10579757 IC50 = 0.01 ug.mL-1 T65755 CAYN96 10597715 IC50 = 40000 nM T65755 C2CQ1X 10627876 IC50 = 86 nM T65755 C3N9BM 10643236 IC50 > 100000 nM T65755 C0KQE7 10651333 IC50 = 1 ug.mL-1 T65755 C9VCT3 10669053 IC50 = 44000 nM T65755 C3KT5X 10707192 IC50 = 811 nM T65755 CK41EV 10746642 IC50 = 330 nM T65755 CQZ36O 10785752 IC50 > 100000 nM T65755 C3FC7X 10800939 IC50 = 2810 nM T65755 CI17AK 10818029 IC50 = 0.065 ug.mL-1 T65755 CD0G3L 10832425 IC50 > 100000 nM T65755 CKS03P 10834447 IC50 = 6000 nM T65755 C4HS8E 10871792 IC50 = 24 nM T65755 C0J5TW 10882720 IC50 = 85000 nM T65755 C9CL4P 10892598 IC50 = 51 nM T65755 CD2O8I 10894419 IC50 = 84 nM T65755 CLQ8S9 10902481 IC50 = 279 nM T65755 CANR41 10914997 IC50 = 67 nM T65755 C0YVZ3 10924497 IC50 = 53000 nM T65755 C37EPU 10925849 IC50 = 30 nM T65755 CS25XQ 10927898 IC50 = 20 nM T65755 C5OUK4 10928349 IC50 = 30 nM T65755 C3HAQ5 10948013 IC50 = 118 nM T65755 CY60KR 10960555 IC50 = 52 nM T65755 CHU31L 10968817 IC50 = 443 nM T65755 CX9C8U 10980767 IC50 = 111 nM T65755 CCT26F 10991689 IC50 = 23 nM T65755 CP2M9H 10999664 IC50 = 5000 nM T65755 CTN9A3 11004308 IC50 = 10 nM T65755 C1BK9H 11014893 IC50 = 164 nM T65755 CKO06G 11022963 IC50 = 2900 nM T65755 C7Y3SH 11024529 IC50 = 23 nM T65755 C7XQ0S 11024550 IC50 = 38 nM T65755 C1RDP4 11024886 IC50 = 37 nM T65755 C30UBP 11025801 IC50 = 278 nM T65755 C3D4CG 11034593 IC50 = 59 nM T65755 CEG9F0 11035042 IC50 = 262 nM T65755 C4I8WQ 11035592 IC50 = 14 nM T65755 C4V6YF 11045824 IC50 = 110000 nM T65755 CQY9K4 11058122 IC50 = 66 nM T65755 CUAT95 11064399 IC50 = 70000 nM T65755 CX50LC 11066195 IC50 = 357 nM T65755 CEPM03 11068867 IC50 = 23 nM T65755 CVWU78 11077840 IC50 = 69 nM T65755 CU87IC 11078239 IC50 = 104000 nM T65755 CAZ08J 11079877 IC50 = 79 nM T65755 CH3M6P 11088199 IC50 = 64 nM T65755 CVC25L 11092030 IC50 = 330 nM T65755 CS7N9U 11111307 IC50 = 40 nM T65755 CB1LI9 11113600 IC50 = 79 nM T65755 CI98LJ 11122087 IC50 = 14 nM T65755 C1XN3B 11129435 IC50 = 36800 nM T65755 C2N8CT 11130223 IC50 = 1000 nM T65755 CFL3D8 11139651 IC50 = 23000 nM T65755 COYG84 11144368 IC50 = 85 nM T65755 C0SJ9A 11149231 IC50 > 100000 nM T65755 C0S1IW 11151102 IC50 = 530 nM T65755 CNCO31 11151694 IC50 = 1100 nM T65755 CAB5Y0 11153120 IC50 > 100000 nM T65755 CYVU80 11162880 IC50 = 130 nM T65755 C0ZF4V 11173451 IC50 = 100 nM T65755 C2KT3W 11173598 IC50 > 100000 nM T65755 CG97FC 11173720 IC50 = 85 nM T65755 CU04YX 11174153 IC50 > 10000 nM T65755 CFZQ65 11176374 IC50 > 100000 nM T65755 C4L0CH 11177533 EC50 = 2100 nM T65755 C0N9RY 11185206 IC50 = 110 nM T65755 C7Z6IS 11186578 IC50 = 820 nM T65755 C9DH5W 11188547 IC50 = 510 nM T65755 C1RMG0 11197404 IC50 > 10000 nM T65755 CZ4J9V 11210392 IC50 < 20000 nM T65755 C8G5WP 11210533 IC50 = 14200 nM T65755 C75MVU 11220440 IC50 < 20000 nM T65755 CNG36U 11220677 IC50 = 84 nM T65755 C9HBY8 11221089 IC50 = 530 nM T65755 C1RTE9 11222711 IC50 < 20000 nM T65755 CWU4V6 11232751 IC50 = 620 nM T65755 CQ41DB 11236322 IC50 = 1200 nM T65755 CA2BV9 11243465 IC50 = 98 nM T65755 C2HVA7 11265575 IC50 = 80000 nM T65755 C40UGT 11265886 IC50 = 79 nM T65755 CS32OD 11269220 IC50 = 4300 nM T65755 C7EZS9 11276149 IC50 = 4270 nM T65755 C69AOS 11277337 IC50 = 670 nM T65755 CDH04Y 11277927 IC50 = 670 nM T65755 CXF3G8 11280414 EC50 = 50 nM T65755 C6FAM0 11280685 IC50 = 74 nM T65755 C60JME 11289208 IC50 > 10000 nM T65755 CMF7L9 11292866 IC50 = 400 nM T65755 CSL7F5 11302073 IC50 = 500 nM T65755 C19SJW 11316731 IC50 = 200 nM T65755 C94SCQ 11324959 IC50 = 210 nM T65755 CDO6U7 11326952 IC50 = 1170 nM T65755 C5J6XT 11335690 IC50 = 660 nM T65755 CA6LJ7 11348920 IC50 = 5200 nM T65755 C0L1BK 11357542 IC50 > 40000 nM T65755 CGUO67 11358869 IC50 = 520 nM T65755 CBZ17A 11359066 IC50 = 230 nM T65755 CMGF30 11360338 IC50 = 172 nM T65755 C8O2KR 11360626 IC50 < 8000 nM T65755 CNY96V 11361410 IC50 = 106 nM T65755 CDS07Y 11362090 EC50 = 420 nM T65755 CIXK40 11362097 IC50 = 220 nM T65755 CFI94W 11369840 IC50 < 80000 nM T65755 CX1UH4 11370046 IC50 > 100000 nM T65755 C0V2DZ 11370695 IC50 = 22000 nM T65755 CB94ZN 11373732 IC50 = 70 nM T65755 C5QH6N 11374190 IC50 = 50 nM T65755 C6HNE4 11379942 IC50 > 10000 nM T65755 CBO37U 11392331 IC50 = 370 nM T65755 CY34EQ 11393847 IC50 = 900 nM T65755 CRH1E9 11403497 IC50 = 350 nM T65755 C3T7SR 11404069 IC50 = 800 nM T65755 CRC21H 11406292 IC50 = 137 nM T65755 C03VUD 11406470 EC50 = 280 nM T65755 CF19EP 11412948 IC50 > 10000 nM T65755 CKD63H 11414031 IC50 = 1600 nM T65755 CP95XA 11414831 IC50 = 1200 nM T65755 C78IKR 11417689 IC50 = 90 nM T65755 C7A5HZ 11420037 IC50 = 569.97 nM T65755 CQRO51 11430433 EC50 = 200 nM T65755 C0TBW6 11430672 IC50 = 590 nM T65755 CQ8DH7 11437795 IC50 < 8000 nM T65755 C4K5JO 11451850 IC50 < 80000 nM T65755 CP7FN8 11460124 IC50 < 8000 nM T65755 CV74KQ 11461551 IC50 = 25 nM T65755 CS2JT5 11462782 IC50 = 570 nM T65755 CH93JP 11470740 IC50 > 100000 nM T65755 CP0V4Z 11483359 IC50 = 941 nM T65755 CL62RB 11483913 IC50 = 3210 nM T65755 CA8I2Z 11485450 IC50 = 80000 nM T65755 CR1C5I 11485984 IC50 = 150 nM T65755 CY34KI 11487392 IC50 = 2600 nM T65755 CEMI96 11490265 IC50 = 2 nM T65755 C10EMT 11492498 IC50 = 788 nM T65755 C24IJH 11494701 IC50 = 1.5 nM T65755 C4INZ5 11501517 EC50 = 460 nM T65755 CK76UT 11507090 IC50 > 25000 nM T65755 CD6V5M 11507610 IC50 = 22 nM T65755 C9E3VI 11509729 EC50 = 26 nM T65755 C7FDW8 11531687 IC50 = 4700 nM T65755 CY91CV 11538378 EC50 = 82 nM T65755 CB3YU1 11545612 IC50 = 1990 nM T65755 C9RT8F 11545665 IC50 = 440 nM T65755 CWCZ73 11547141 IC50 = 15000 nM T65755 C3JK5A 11551699 IC50 = 3500 nM T65755 CO53NI 11551748 IC50 = 55830 nM T65755 C5XHP3 11552702 EC50 = 1500 nM T65755 CIV4D2 11554742 IC50 = 3200 nM T65755 CM1IP7 11557720 IC50 > 25000 nM T65755 CS6HM3 11558091 IC50 = 2800 nM T65755 C2F9NT 11558827 IC50 = 700 nM T65755 C0QY4A 11560153 EC50 = 59 nM T65755 CDV3R4 11562023 IC50 = 89680 nM T65755 C3UL7I 11572286 IC50 > 100000 nM T65755 CJEU40 11573286 IC50 = 188 nM T65755 CWV81D 11574525 EC50 = 850 nM T65755 CM4LE6 11581475 IC50 = 2 nM T65755 C08SKT 11583320 IC50 = 160 nM T65755 COL83R 11588699 EC50 = 950 nM T65755 CPM18I 11593830 IC50 = 1700 nM T65755 CLDP05 11597343 IC50 = 1600 nM T65755 C8HL7A 11603909 IC50 = 550 nM T65755 CGX9Q4 11604452 EC50 = 1000 nM T65755 CY3EQ1 11609655 IC50 > 100000 nM T65755 C73VWD 11621069 IC50 = 96260 nM T65755 C23LRB 11623126 IC50 = 11000 nM T65755 CP78NE 11625086 EC50 = 170 nM T65755 CTK52W 11625292 EC50 = 47 nM T65755 CY2E7K 11631108 IC50 > 100000 nM T65755 CK73QE 11638839 EC50 = 330 nM T65755 CU4OM8 11638926 IC50 = 1.7 nM T65755 CX0S1Z 11639772 EC50 = 88 nM T65755 CL3PS9 11639915 EC50 = 29 nM T65755 C6SNG5 11649112 IC50 = 84400 nM T65755 C9RD5U 11651487 IC50 = 252 nM T65755 CG5XV9 11667696 EC50 = 100 nM T65755 CP4DR5 11670005 IC50 = 11000 nM T65755 CG9OC4 11682502 IC50 = 1.05 nM T65755 CHM8S1 11687325 IC50 = 302 nM T65755 C1N2TG 11688241 IC50 = 8600 nM T65755 C5W1FX 11688802 IC50 = 32000 nM T65755 C70WUT 11690588 EC50 = 790 nM T65755 CT9O2D 11691923 IC50 = 66110 nM T65755 CMG97J 11696043 IC50 = 56400 nM T65755 CH4GE5 11696917 EC50 = 67100 nM T65755 C32CFI 11696935 IC50 = 83660 nM T65755 C3U2IC 11697190 EC50 = 280 nM T65755 CBV1O8 11703489 IC50 = 10400 nM T65755 C4VM0G 11704283 EC50 = 11200 nM T65755 C7W4OF 11704469 EC50 = 100 nM T65755 CD3MV8 11705012 EC50 = 4300 nM T65755 C2VU8O 11712658 IC50 = 46800 nM T65755 C3CD8P 11722754 IC50 = 359 nM T65755 CC1SD4 11722988 IC50 = 6000 nM T65755 CX2GR8 11723098 IC50 = 100 nM T65755 C4JWU0 11730819 IC50 = 370 nM T65755 C19LDJ 11737664 IC50 = 230000 nM T65755 CR3DP5 11738326 IC50 = 5000 nM T65755 CH8J4L 11759466 IC50 = 46 nM T65755 C1T7NO 11760982 IC50 = 24 nM T65755 C28AFE 11783488 IC50 = 27 nM T65755 CH57PG 11783698 IC50 = 53 nM T65755 C9Y2GM 11794739 IC50 > 100000 nM T65755 C58FZA 11795873 IC50 = 7700 nM T65755 C5V6FM 11810219 IC50 = 53 nM T65755 CQX1J0 11810423 IC50 = 220 nM T65755 C6XQN8 11817924 IC50 = 150000 nM T65755 CQ5WH8 11818464 IC50 = 7500000 nM T65755 C83ZIK 11848284 EC50 = 30 nM T65755 CN2R1O 11848285 EC50 = 500 nM T65755 CRD85U 11848286 EC50 = 30 nM T65755 C3TVQ7 11848287 EC50 = 380 nM T65755 CEOI97 11848476 EC50 = 200 nM T65755 CQ0A2T 11848478 EC50 = 3270 nM T65755 CFSG39 11848898 IC50 = 173 nM T65755 CG4M0H 11848899 IC50 = 124 nM T65755 CL2P8T 11848948 IC50 = 128 nM T65755 C6J4KH 11848949 IC50 = 181 nM T65755 CE5I9U 11849152 EC50 = 1300 nM T65755 CB61ZA 11849153 EC50 = 430 nM T65755 CRM5E9 11849154 EC50 = 150 nM T65755 CRIS81 11849155 EC50 = 840 nM T65755 CL19WI 11849156 EC50 = 340 nM T65755 CU0M1E 11947684 IC50 = 1 nM T65755 CWR4Q9 11957768 IC50 = 1.5 nM T65755 CF06BI 11963978 IC50 = 15 nM T65755 C5LNX0 12000743 IC50 = 46400 nM T65755 CJQ8L0 12001305 IC50 = 7.2 nM T65755 CIT53J 12291400 IC50 = 135 nM T65755 C9D8FE 12988035 IC50 = 1680 nM T65755 CO5A0Q 12988036 IC50 = 524 nM T65755 CCDO27 13735499 IC50 = 71000 nM T65755 C4XJ8M 13889849 IC50 = 430 nM T65755 CS6B0L 14067176 IC50 = 501.19 nM T65755 CP1OD5 14452250 IC50 = 100000 nM T65755 CH48FC 15399275 IC50 = 600 nM T65755 CC45ME 15484557 IC50 = 419 nM T65755 C9QY2A 15484558 IC50 = 257 nM T65755 CVX5J4 15484559 IC50 = 4 nM T65755 CPB9S3 15721949 IC50 = 125.89 nM T65755 CS1QO9 15986509 IC50 = 8700 nM T65755 CK0R6X 16051663 EC50 = 240 nM T65755 CE7TC8 16051665 EC50 = 95 nM T65755 CG37SA 16051667 EC50 = 360 nM T65755 C7NVE6 16051775 EC50 = 150 nM T65755 C9ZQB3 16095102 IC50 = 45 nM T65755 C80XYC 16095113 IC50 = 1300 nM T65755 C6RE2F 16220721 Ki = 13.67 nM T65755 C09FZM 16220753 IC50 = 167 nM T65755 CG87WA 16655008 IC50 = 3.8 nM T65755 CEXS90 16720330 IC50 > 10000 nM T65755 CPD20L 16720331 IC50 = 270 nM T65755 C90FCL 16720547 IC50 > 10000 nM T65755 CUG50I 16733294 IC50 = 80 nM T65755 CV54SY 16733414 IC50 = 900 nM T65755 CBF9Z0 16739374 IC50 = 72000 nM T65755 C7ORU3 17754279 EC50 = 44 nM T65755 CWF1J8 17754282 EC50 = 110 nM T65755 CU23ZA 17754370 EC50 = 67 nM T65755 C4PNK7 17754416 EC50 = 190 nM T65755 C1N8UM 17754469 EC50 = 220 nM T65755 C2CKX5 17754471 EC50 = 53 nM T65755 C4S6RU 17754512 EC50 = 220 nM T65755 C0KA9P 17754513 EC50 = 44 nM T65755 CW76MC 17754514 EC50 = 110 nM T65755 CZTA06 17754556 EC50 = 61 nM T65755 CAJ0S2 17754557 EC50 = 25 nM T65755 C89RLB 17754559 EC50 = 29 nM T65755 CWBN48 17754922 EC50 = 38 nM T65755 C5NTU2 17754923 EC50 = 160 nM T65755 CCU15F 17754925 EC50 = 91 nM T65755 CA5RT9 17755228 EC50 = 2650 nM T65755 CZ79PM 17756301 IC50 = 270 nM T65755 CT7K6N 17756302 IC50 = 260 nM T65755 C9MNR8 17756303 EC50 = 1000 nM T65755 CU4E3H 17756304 IC50 = 310 nM T65755 CC2GS4 17756305 EC50 = 4270 nM T65755 CF7JR0 17756401 IC50 = 39 nM T65755 CPVI84 17756402 EC50 = 1100 nM T65755 C3FN8M 17756403 EC50 = 290 nM T65755 C5YS2I 17756404 EC50 = 2670 nM T65755 C63DPZ 17756405 IC50 = 120 nM T65755 CY1V6H 17756406 IC50 = 340 nM T65755 C8GBK4 17756407 EC50 = 2570 nM T65755 CZ1P9D 17756505 EC50 = 4100 nM T65755 C8G9FC 17756506 IC50 = 1000 nM T65755 CDY7R2 20655275 IC50 = 73100 nM T65755 C9UX2V 20785858 IC50 < 200 nM T65755 CV8QU0 21581855 IC50 = 44 nM T65755 CX57LO 21670609 IC50 = 0.3 nM T65755 C61KUX 21726402 IC50 > 40 nM T65755 C0SMZ1 23072426 EC50 = 25000 nM T65755 C9O5EB 23072489 EC50 = 15000 nM T65755 C3Z2EA 23092216 IC50 = 141 nM T65755 C5YHP3 23092284 IC50 = 46 nM T65755 C27ECN 23092286 IC50 = 101 nM T65755 CJAT82 23557362 IC50 > 100000 nM T65755 CEF8W4 23625604 IC50 = 375 nM T65755 C5RO8F 23625605 IC50 = 398.11 nM T65755 COL1C3 23625606 IC50 = 199.53 nM T65755 C36NKL 23648268 IC50 = 150 nM T65755 CH35NV 23656767 IC50 = 242 nM T65755 C0VXI8 23657111 IC50 > 3200 nM T65755 CE85CP 23657268 IC50 = 7 nM T65755 CU01QJ 24178404 IC50 = 3.9 nM T65755 CQN7X0 24186135 IC50 = 198000 nM T65755 C8RC9P 24744325 Ki = 16 nM T65755 CH35QK 24748984 IC50 = 14000 nM T65755 CYG18K 24748985 IC50 = 20100 nM T65755 C6M4QN 24748986 IC50 = 60 nM T65755 CK32AR 24749071 IC50 = 10400 nM T65755 C9E0AU 24749072 IC50 > 100000 nM T65755 C7Z5JT 24756560 IC50 = 226 nM T65755 COWH36 24756635 IC50 = 186 nM T65755 CYTH62 24756636 IC50 = 280 nM T65755 CDZ4K7 24756711 IC50 = 350 nM T65755 CTU6C9 24756884 IC50 = 175 nM T65755 CJ2ZV1 24756885 IC50 = 141 nM T65755 CJ3FB0 24756886 IC50 = 30 nM T65755 CKG92U 24756975 IC50 = 12 nM T65755 CE84QS 24757061 IC50 = 27 nM T65755 CJ3RD8 24757063 IC50 = 53 nM T65755 C3GY1L 24757860 IC50 = 183 nM T65755 CBI16V 24779712 IC50 = 37 nM T65755 C0YKE4 24779713 IC50 = 30 nM T65755 C4N6PA 24854436 IC50 = 3800 nM T65755 CR10WY 24854582 IC50 = 4900 nM T65755 CI3B6L 24857909 EC50 = 12000 nM T65755 CPU1Z5 24893969 IC50 = 83 nM T65755 CP29ZE 24893970 IC50 = 120 nM T65755 CHKZ02 24894417 IC50 = 3410 nM T65755 C6BNX7 24894418 IC50 = 115 nM T65755 CQ63WU 24894419 IC50 = 467 nM T65755 C3E0SN 24894423 IC50 = 630.96 nM T65755 CA56SQ 24894517 IC50 = 719 nM T65755 CVA4J1 24894518 IC50 = 87 nM T65755 C7FV6W 24894519 IC50 = 386 nM T65755 C8R2KN 24894520 IC50 = 384 nM T65755 C2EQS1 24894522 IC50 = 1230 nM T65755 CJWI39 24894523 IC50 = 74 nM T65755 CJ15OF 24894524 IC50 = 74 nM T65755 CKQZ25 24894639 IC50 = 42 nM T65755 CITS83 24894640 IC50 = 646 nM T65755 CX3QD8 24894641 IC50 = 174 nM T65755 CC1G2E 24894642 IC50 = 748 nM T65755 CJ64TA 24894643 IC50 = 1500 nM T65755 C1PTW8 24894644 IC50 = 500 nM T65755 CKJC01 24894645 IC50 = 32 nM T65755 CW3MP6 24894775 IC50 = 79 nM T65755 C6YL4C 24894776 IC50 = 25 nM T65755 CA2O6T 24894777 IC50 = 16 nM T65755 C8XS0N 24894778 IC50 = 15 nM T65755 C6CK9N 24894779 IC50 = 97 nM T65755 CXY5C7 24894780 IC50 = 19 nM T65755 CT4RJ0 24894895 IC50 = 15 nM T65755 CJTP74 24894896 EC50 = 2400 nM T65755 C4F5TN 24894897 EC50 = 760 nM T65755 C75WEJ 24894898 IC50 = 2990 nM T65755 CMT7F4 24894899 IC50 = 36 nM T65755 CH13WV 24894900 IC50 = 49 nM T65755 CA5V7S 24894901 IC50 = 46 nM T65755 CDU08E 24895004 IC50 = 40 nM T65755 C1IR2A 24895005 IC50 = 8 nM T65755 CQJ78L 24895006 IC50 = 48 nM T65755 C4PN6I 24895007 IC50 = 110 nM T65755 C9H1WI 24895008 IC50 = 14 nM T65755 CYM91Q 24895009 IC50 = 49 nM T65755 CEH9A4 24895010 IC50 = 423 nM T65755 C8SP7C 24895115 IC50 = 26 nM T65755 C0C9VU 24895116 IC50 = 18 nM T65755 CM3Q7A 24895117 IC50 = 8 nM T65755 CZ1SP9 24895118 IC50 = 195 nM T65755 CY7D1N 24895120 IC50 = 128 nM T65755 CH7L8Z 24895121 IC50 = 293 nM T65755 C60FAX 24895122 IC50 = 94 nM T65755 CO68DV 24895187 IC50 = 6590 nM T65755 C40QJO 24895188 IC50 = 1995.26 nM T65755 C2K8BR 24895189 IC50 = 1480 nM T65755 CBI25A 24895190 IC50 = 127 nM T65755 C96GPD 24944848 IC50 = 40900 nM T65755 CNMB03 24944849 IC50 > 100000 nM T65755 CTCB27 24944850 IC50 = 551 nM T65755 C5PH0N 24944851 IC50 = 31 nM T65755 CK17HZ 24944855 IC50 = 34.1 nM T65755 C0BOJ2 24944856 IC50 = 66.6 nM T65755 CX05SV 24944930 IC50 = 6.5 nM T65755 CB8EZ0 24944934 IC50 = 421 nM T65755 C2CP6T 24944935 IC50 = 13.2 nM T65755 C1NZ8X 24945115 IC50 = 4.4 nM T65755 CF0U4T 24945204 IC50 = 8.4 nM T65755 C8W3YA 24945368 IC50 = 15.3 nM T65755 C2MYN7 24945689 IC50 = 58.1 nM T65755 CRPM36 25014636 IC50 = 14.2 nM T65755 C82REW 25014637 IC50 = 9.6 nM T65755 C8ZVO2 25014638 IC50 = 67.6 nM T65755 CDBZ21 25014718 IC50 = 1.8 nM T65755 C5B0IJ 25023793 IC50 = 380 nM T65755 CLG23N 25023794 IC50 = 3.7 nM T65755 C9BK7U 25023852 IC50 = 5888.44 nM T65755 CZP26Q 25023853 IC50 = 26915.35 nM T65755 CD04RS 25067623 IC50 = 365.8 nM T65755 CUWG27 25067624 IC50 = 15.9 nM T65755 CIR82T 25067628 IC50 = 425.8 nM T65755 CIG6U8 25068424 IC50 = 363.6 nM T65755 CB2U1I 25068428 IC50 = 4.3 nM T65755 C5GNP0 25068480 IC50 = 52.4 nM T65755 C2U0VC 25068481 IC50 = 2.09 nM T65755 CF7NR1 25068482 IC50 = 287.2 nM T65755 CO1L7Y 25068483 IC50 = 106.1 nM T65755 C3A2FO 25118057 IC50 = 340 nM T65755 CFS5O4 25168576 EC50 = 6500 nM T65755 C1MTJ3 25183354 IC50 = 15 nM T65755 CP6HD4 25206847 IC50 = 87 nM T65755 C71BSC 25206848 IC50 = 20 nM T65755 CGT40Q 25206850 IC50 = 74 nM T65755 CZW74M 25206851 IC50 = 24 nM T65755 CF4W5Z 25206852 IC50 = 27 nM T65755 CU9QE0 25207011 IC50 = 17 nM T65755 C9RSJ1 25207012 IC50 = 33 nM T65755 CRLK27 25207013 IC50 = 53 nM T65755 CUN37O 25207014 IC50 = 32 nM T65755 C5DOJ4 25207016 IC50 = 56 nM T65755 C7Q9SI 25207163 IC50 = 41 nM T65755 CB29PE 25211681 EC50 = 600 nM T65755 C2YG9N 25216677 IC50 > 50000 nM T65755 C5CZV0 25216678 IC50 = 4900 nM T65755 CB6C2A 25216810 IC50 = 7200 nM T65755 CPX03T 25217055 IC50 > 50000 nM T65755 CP26WM 25217056 IC50 = 9900 nM T65755 CBDR02 25217057 IC50 = 9500 nM T65755 C9URH7 25217288 IC50 = 6400 nM T65755 C2WH9J 25217398 IC50 > 50000 nM T65755 CSM0F2 25217513 IC50 = 180 nM T65755 CU53WB 42596953 IC50 = 47 nM T65755 C8OQ0G 42598944 IC50 = 28 nM T65755 C2LES7 42599455 IC50 = 23 nM T65755 C2KO0F 42599456 IC50 = 9 nM T65755 CK3OM4 42599457 IC50 = 25 nM T65755 CO6AI7 42599458 IC50 = 20 nM T65755 CC5BY2 42599459 IC50 = 21 nM T65755 C82ELT 42599709 IC50 = 338 nM T65755 C5UH4B 42601409 IC50 = 1190 nM T65755 C3P6NY 42601488 IC50 = 620 nM T65755 COI7Y3 42611300 IC50 = 19 nM T65755 CU23PG 42611301 IC50 < 1 nM T65755 C62QFJ 42611486 IC50 = 40 nM T65755 CLH2Q7 42612852 IC50 = 324 nM T65755 C7GIQ3 42625508 EC50 = 1710 nM T65755 CVZ83M 42625582 EC50 = 3380 nM T65755 C5MD9E 42625892 EC50 = 1600 nM T65755 CCJ3O7 42637070 IC50 = 1200 nM T65755 C4P2JM 42637074 IC50 = 4400 nM T65755 C2FS9H 42637148 IC50 > 100000 nM T65755 C5LZ8W 42637149 IC50 = 16000 nM T65755 CDP49E 42637220 IC50 > 100000 nM T65755 CAG92C 42637221 IC50 > 100000 nM T65755 C53UQX 42637222 IC50 > 100000 nM T65755 CM80NB 42637223 IC50 > 100000 nM T65755 CT9X5J 42637224 IC50 > 100000 nM T65755 C96CZE 42637225 IC50 = 2000 nM T65755 C7IZN8 42637295 IC50 = 13000 nM T65755 C8EZF3 42637296 IC50 = 1400 nM T65755 CX95OH 42637297 IC50 = 11000 nM T65755 CO3V1N 42637298 IC50 = 30000 nM T65755 CB79DG 42637299 IC50 = 1600 nM T65755 CP36KB 42637300 IC50 = 17000 nM T65755 CI8J6H 42637372 IC50 = 920 nM T65755 C5RYO0 42637373 IC50 = 24000 nM T65755 C6M7EY 42637790 IC50 = 12000 nM T65755 C6ZFH7 42637791 IC50 = 23000 nM T65755 CWM68Z 42637850 IC50 > 100000 nM T65755 CE75UJ 42637851 IC50 > 100000 nM T65755 CF6A5E 42637852 IC50 > 100000 nM T65755 C4IJY2 42637853 IC50 = 4200 nM T65755 CUMF52 42637854 IC50 = 2000 nM T65755 C0I2AP 42637855 IC50 = 4700 nM T65755 C6CNV4 42637926 IC50 > 100000 nM T65755 C53JDS 42637927 IC50 = 51000 nM T65755 CJ0CG5 42638004 IC50 = 15000 nM T65755 C8X0TG 42638005 IC50 = 1400 nM T65755 C4JU1S 42642257 IC50 = 10000 nM T65755 CA80MF 42642258 IC50 = 10 nM T65755 CEP8Z7 42642259 IC50 = 100000 nM T65755 C97JKT 42642260 IC50 = 918700 nM T65755 C21RGW 42642262 IC50 = 80 nM T65755 CRA12H 42642371 IC50 = 250 nM T65755 CAG5L0 44228659 IC50 = 42 nM T65755 CPD6S7 44240793 IC50 = 82 nM T65755 CY0QB9 44253226 IC50 = 100 nM T65755 CAD81N 44253358 IC50 = 641 nM T65755 C7HID9 44253359 IC50 = 316 nM T65755 CG2YN5 44253360 IC50 = 288 nM T65755 C6T8VW 44253361 IC50 = 140 nM T65755 CX3FV8 44253363 IC50 = 1410 nM T65755 C1KGP6 44253364 IC50 = 2173 nM T65755 CJB5N8 44253504 IC50 = 1040 nM T65755 CR6MQ7 44253505 IC50 = 366 nM T65755 CF9TP8 44253506 IC50 = 408 nM T65755 CRC12W 44253507 IC50 = 9020 nM T65755 CY96UN 44253508 IC50 = 1210 nM T65755 CZ1A8P 44253509 IC50 = 1190 nM T65755 COI6B0 44253648 IC50 = 5150 nM T65755 CE30GS 44253652 IC50 = 221 nM T65755 CE8UP5 44253653 IC50 = 932 nM T65755 CN2C6P 44253777 IC50 > 50000 nM T65755 CJU49N 44253778 IC50 = 2550 nM T65755 CX24QL 44253779 IC50 = 2990 nM T65755 CZ8R1N 44253780 IC50 = 83 nM T65755 CW3U7O 44299072 IC50 = 41 nM T65755 CO0JI5 44299073 IC50 = 56.5 nM T65755 CPG8J9 44299082 IC50 = 80.3 nM T65755 C1LAT5 44299123 IC50 = 15 nM T65755 C14MQD 44299132 IC50 = 31.4 nM T65755 C5T9SX 44299141 IC50 = 15 nM T65755 C0BTW5 44299150 IC50 = 37.5 nM T65755 CC59YB 44299365 IC50 = 3.1 nM T65755 C1S0OQ 44299378 IC50 = 5.4 nM T65755 CU7Q1P 44299423 IC50 = 732 nM T65755 C5B8DA 44299452 IC50 = 3.5 nM T65755 CSPK87 44299473 IC50 = 6.5 nM T65755 C3QLV4 44299474 IC50 = 3.1 nM T65755 CZWC71 44322089 IC50 = 80000 nM T65755 C3GJ2X 44322091 IC50 = 61000 nM T65755 C80TRE 44322612 IC50 = 30000 nM T65755 CW3D8V 44328913 EC50 = 10000 nM T65755 C6RLC5 44328915 EC50 = 10000 nM T65755 C6AUY0 44328918 EC50 = 10000 nM T65755 C8R4IO 44328919 EC50 = 5000 nM T65755 C86IOC 44328927 EC50 = 3000 nM T65755 C1NL0Q 44328959 EC50 = 3000 nM T65755 C9C5VS 44328965 EC50 = 3000 nM T65755 C4ER7O 44328966 EC50 > 25000 nM T65755 CC8OK4 44328974 EC50 = 99000 nM T65755 C96CLW 44328975 EC50 = 10000 nM T65755 CH7VS1 44329159 EC50 = 20000 nM T65755 CK6NG2 44329200 EC50 = 25000 nM T65755 C2O7MW 44329201 EC50 = 2000 nM T65755 C42PYJ 44329220 EC50 = 5000 nM T65755 CX5HB8 44330308 IC50 = 1.4 nM T65755 C8OD2I 44330309 IC50 = 660 nM T65755 C1UTD8 44330464 IC50 = 2.1 nM T65755 CZ9IT6 44330499 IC50 = 99 nM T65755 CGXL80 44330508 IC50 = 38 nM T65755 CG7Q2D 44330512 IC50 > 5000 nM T65755 C72KRD 44330513 IC50 = 640 nM T65755 CB16KI 44330551 IC50 = 66 nM T65755 C37UZK 44330590 IC50 = 5000 nM T65755 C7YLS5 44340625 IC50 > 100000 nM T65755 CYB0V6 44340841 IC50 > 50000 nM T65755 CV73WM 44340857 IC50 = 4900 nM T65755 CB7OA9 44340858 IC50 > 50000 nM T65755 CR8Y4A 44341042 IC50 > 5000 nM T65755 C1ZTO5 44341043 IC50 = 110 nM T65755 CHA48J 44341044 IC50 = 109 nM T65755 CB79UK 44341045 IC50 = 62 nM T65755 CW9BU1 44341230 IC50 > 50000 nM T65755 CAUH13 44341243 IC50 = 82 nM T65755 CSDN36 44341245 IC50 = 3.1 nM T65755 C0M7UH 44342832 IC50 = 8600 nM T65755 CNR9L1 44342955 IC50 = 16000 nM T65755 CL0R4X 44342956 IC50 = 3000 nM T65755 CJLK34 44342958 IC50 = 2200 nM T65755 CD3N9B 44342959 IC50 > 50000 nM T65755 C1QF2Y 44343064 IC50 = 3200 nM T65755 CUYA48 44343093 IC50 > 50000 nM T65755 CO45AJ 44343096 IC50 = 2900 nM T65755 C56VJE 44349482 IC50 = 2.7 nM T65755 CFZB27 44349491 IC50 = 4.4 nM T65755 C03MFI 44349504 IC50 = 5.8 nM T65755 CDO6W9 44349514 IC50 = 74 nM T65755 CC6X1U 44349632 IC50 = 9.8 nM T65755 CFY03T 44349683 IC50 = 4.3 nM T65755 C67GVD 44349684 IC50 = 4.3 nM T65755 CBA2P4 44349738 IC50 = 42 nM T65755 C2L8DG 44349739 IC50 = 11 nM T65755 CPH7L0 44349740 IC50 = 8.5 nM T65755 C0ZK9R 44349758 IC50 = 2.5 nM T65755 C5CYS2 44349760 IC50 = 23 nM T65755 C0B9GZ 44349778 IC50 = 12 nM T65755 CA2VX5 44349782 IC50 = 19 nM T65755 CZ3AE7 44349795 IC50 = 89 nM T65755 CS2ZP1 44349814 IC50 = 13 nM T65755 CAL45Y 44350633 IC50 = 1800 nM T65755 CHCA36 44350642 IC50 = 340 nM T65755 C0EK1O 44350643 IC50 = 90 nM T65755 CZ7DS3 44350659 IC50 > 50000 nM T65755 CVX13P 44350680 IC50 > 50000 nM T65755 CH0ZE6 44350681 IC50 > 50000 nM T65755 C01QIX 44350686 IC50 = 610 nM T65755 CUM4X7 44350687 IC50 = 540 nM T65755 CV4WT2 44350688 IC50 = 250 nM T65755 CM6W4L 44350719 IC50 = 430 nM T65755 CX27QF 44350720 IC50 > 50000 nM T65755 CN1LI6 44350775 IC50 > 50000 nM T65755 CO1C9T 44350784 IC50 > 50000 nM T65755 C8BO6C 44350785 IC50 > 50000 nM T65755 CS4K5H 44350789 IC50 = 1830 nM T65755 CEX41R 44350797 IC50 = 1500 nM T65755 C0ZUG8 44350805 IC50 > 10000 nM T65755 C07VMF 44350808 IC50 = 580 nM T65755 CM6B3H 44350811 IC50 = 6400 nM T65755 CZ42BY 44350825 IC50 = 310 nM T65755 C9AEI5 44351006 IC50 = 320 nM T65755 CN41AE 44351010 IC50 > 50000 nM T65755 CY0BK8 44351018 IC50 > 50000 nM T65755 C3BAE8 44356874 IC50 = 121000 nM T65755 C7WD0R 44356939 IC50 > 1000000 nM T65755 CJ64OF 44356966 IC50 > 100000 nM T65755 CYV76I 44356975 IC50 > 100000 nM T65755 CTAL56 44356976 IC50 > 100000 nM T65755 CF2UW5 44357041 IC50 > 100000 nM T65755 CY8IN4 44357083 IC50 = 650000 nM T65755 CJ3F6G 44357100 IC50 = 300000 nM T65755 C0HPU2 44357121 IC50 > 100000 nM T65755 CC1WV5 44357122 IC50 > 100000 nM T65755 CE8S3K 44357123 IC50 > 100000 nM T65755 C0U3IO 44357182 IC50 > 100000 nM T65755 CX61RT 44357183 IC50 > 100000 nM T65755 CU2HM6 44357407 IC50 > 100000 nM T65755 C0C3EA 44357425 IC50 > 100000 nM T65755 C7G5CO 44359547 IC50 = 4000 nM T65755 CIT7A9 44359548 IC50 > 100000 nM T65755 CUM0Q6 44359555 IC50 = 50000 nM T65755 CQ7J2G 44359674 IC50 = 2800 nM T65755 C2V4DN 44359681 IC50 = 4400 nM T65755 CQ5Y8G 44359800 IC50 > 100000 nM T65755 C7C3PR 44365075 IC50 = 5000 nM T65755 C85LYZ 44365258 IC50 = 29.6 nM T65755 CA7SU0 44377463 IC50 > 10000 nM T65755 CU45ZH 44389573 IC50 = 900 nM T65755 CBC4O5 44392266 IC50 = 24000 nM T65755 CDR94X 44392304 IC50 = 3000 nM T65755 C1O6WE 44400358 IC50 = 30 nM T65755 CO6S4D 44401338 IC50 = 70000 nM T65755 CT5KU1 44401387 IC50 = 2500 nM T65755 C1F3HD 44401388 IC50 = 2350 nM T65755 CPI5C2 44401484 IC50 = 2800 nM T65755 C0LAP5 44401548 IC50 = 3100 nM T65755 CJE47N 44401572 IC50 = 1500 nM T65755 CS2DT5 44401640 IC50 = 10200 nM T65755 CD4EC2 44401641 IC50 = 39500 nM T65755 CEO3Q8 44404200 EC50 = 407 nM T65755 C5U9SV 44406761 IC50 = 9400 nM T65755 C5ZX0J 44418116 IC50 = 5 nM T65755 CMK6D5 44418152 IC50 = 9 nM T65755 C5MVF9 44418166 IC50 = 34 nM T65755 C6IBO4 44418169 IC50 = 13 nM T65755 CU37ON 44418170 IC50 = 107 nM T65755 CT81MK 44418184 IC50 = 8 nM T65755 CV0I5E 44418191 IC50 = 5 nM T65755 CTN6G4 44418194 IC50 = 22 nM T65755 CT2DL9 44418195 IC50 = 20 nM T65755 CJAB06 44418207 IC50 = 6 nM T65755 CQ08NE 44427329 IC50 = 398.11 nM T65755 C6ENC3 44427332 IC50 = 375 nM T65755 CP64QU 44427333 IC50 = 1258.93 nM T65755 CQI4O3 44427334 IC50 = 251.19 nM T65755 CEIX21 44427336 IC50 = 316.23 nM T65755 CSB7L1 44427337 IC50 = 100 nM T65755 CN0CL8 44427339 IC50 = 79.43 nM T65755 C0DQC7 44427340 IC50 = 100 nM T65755 CXW6K0 44427341 IC50 = 100 nM T65755 CY01WJ 44427342 IC50 = 50.12 nM T65755 C80BVD 44427343 IC50 = 39.81 nM T65755 CEY1S0 44427344 IC50 = 2511.89 nM T65755 C6RU3C 44427346 IC50 = 1995.26 nM T65755 CP2CU4 44427347 IC50 = 1000 nM T65755 CRYS09 44427348 IC50 = 1258.93 nM T65755 CQ27OM 44427350 IC50 = 3981.07 nM T65755 CO0U4M 44427353 IC50 = 501.19 nM T65755 CO3DC8 44427354 IC50 = 31622.78 nM T65755 C2ZCK9 44427355 IC50 = 501.19 nM T65755 C3G6JH 44427356 IC50 = 501.19 nM T65755 CC0Q6Y 44427358 IC50 = 794.33 nM T65755 C8J3XD 44427359 IC50 = 630.96 nM T65755 C3VP4O 44427360 IC50 = 1995.26 nM T65755 CI23OZ 44431491 IC50 = 134000 nM T65755 C9X3GI 44431493 IC50 = 449000 nM T65755 C61NOW 44431496 IC50 = 154000 nM T65755 C1DH6S 44431497 IC50 = 144000 nM T65755 C7KJV9 44431498 IC50 = 87000 nM T65755 C5YRC9 44431499 IC50 = 226000 nM T65755 CR56OK 44440675 IC50 = 76130 nM T65755 CXA2O0 44443377 IC50 = 2970 nM T65755 CWD74J 44443378 IC50 = 1900 nM T65755 CQS9A7 44443380 IC50 = 2100 nM T65755 C6N3JO 44443381 IC50 = 860 nM T65755 CYQ27L 44443386 IC50 = 1940 nM T65755 C30RIH 44443388 IC50 = 440 nM T65755 C0YS4H 44443393 IC50 = 560 nM T65755 CRO8K7 44443399 IC50 = 450 nM T65755 CE4QS2 44443405 IC50 = 230 nM T65755 C2UF0D 44443412 IC50 = 320 nM T65755 C60CDO 44443416 IC50 = 270 nM T65755 CZNP93 44443418 IC50 = 200 nM T65755 CL2C5H 44443419 IC50 = 110 nM T65755 CQ05RE 44449235 IC50 = 36307.81 nM T65755 C5K7LA 44449588 IC50 = 58 nM T65755 C2ZWV0 44452860 IC50 = 2000 nM T65755 C7N5PQ 44453388 IC50 = 17500 nM T65755 CRQ4L0 44453452 IC50 > 10000 nM T65755 C58YCH 44456972 IC50 > 40000 nM T65755 CE4ZA6 44456992 IC50 = 4.3 nM T65755 CY4I7R 44456994 IC50 = 13300 nM T65755 C5HS2K 44456995 IC50 > 10000 nM T65755 CZR93G 44457014 IC50 = 140 nM T65755 C1B5QO 44457015 IC50 = 96 nM T65755 CM95VA 44457016 IC50 = 150 nM T65755 C1D6IS 44457072 IC50 = 18 nM T65755 CD4V0T 44457073 IC50 = 15 nM T65755 CNS0B6 44457074 IC50 = 128 nM T65755 C9M3OQ 44457097 IC50 = 9 nM T65755 C3Y6IZ 44457098 IC50 = 146 nM T65755 C1FWD0 44457100 IC50 = 19 nM T65755 CTEU41 44457127 IC50 = 1000 nM T65755 C4Y7HG 44457128 IC50 = 700 nM T65755 CY73GA 44457145 IC50 = 800 nM T65755 C3UV7C 44561976 IC50 = 630 nM T65755 CU92TP 44562080 IC50 = 1890 nM T65755 CTUG48 44568433 IC50 = 44 nM T65755 CQT05D 44571772 EC50 = 150 nM T65755 CEZC26 44571987 EC50 = 150 nM T65755 C1EPF2 44571988 EC50 = 42 nM T65755 CUO3V0 44572289 IC50 = 17000 nM T65755 CFH95O 44572348 IC50 = 18000 nM T65755 CD17KA 44572349 IC50 = 19000 nM T65755 CU4VC9 44572350 IC50 = 9100 nM T65755 C5TBI9 44572351 IC50 = 3600 nM T65755 COM65J 44572384 EC50 = 2350 nM T65755 CV91YE 44572385 EC50 = 1040 nM T65755 CAUH07 44572405 IC50 > 50000 nM T65755 CUO41X 44572406 IC50 = 530 nM T65755 CY0I4X 44572407 IC50 = 3200 nM T65755 C3CB2K 44572429 EC50 = 3900 nM T65755 CM2Q8J 44572430 EC50 = 2600 nM T65755 C8AO6P 44572466 IC50 = 3200 nM T65755 C2O3IS 44572467 IC50 > 50000 nM T65755 CH09QJ 44572468 IC50 = 6800 nM T65755 CMAT21 44572489 EC50 = 1150 nM T65755 CU1SY9 44572490 EC50 = 1470 nM T65755 CSD74G 44572491 EC50 = 1700 nM T65755 CZ2X7L 44572516 IC50 = 6100 nM T65755 CW7BK3 44572517 IC50 > 50000 nM T65755 C59TVW 44572518 IC50 = 29000 nM T65755 CC74WS 44572519 IC50 = 38000 nM T65755 CA9WO3 44572537 EC50 = 3000 nM T65755 C06SLW 44572538 EC50 = 1740 nM T65755 CY8TG3 44572539 EC50 = 460 nM T65755 C1JR4C 44572540 EC50 = 7800 nM T65755 CV50NO 44572558 IC50 = 590 nM T65755 CB9Z4E 44572559 IC50 = 12000 nM T65755 C0RUB9 44572560 IC50 = 5800 nM T65755 CZ0PA9 44572581 EC50 = 4400 nM T65755 CD9VR5 44572582 EC50 = 1500 nM T65755 CG5UK0 44572584 EC50 = 1010 nM T65755 CMX32U 44572633 EC50 = 2800 nM T65755 CA3UR6 44572654 IC50 = 2200 nM T65755 C93GWB 44583037 IC50 = 36 nM T65755 CB0J2U 44583049 IC50 = 62 nM T65755 C84PJY 44585257 IC50 = 13.9 nM T65755 C4X7KR 44585258 IC50 = 76 nM T65755 CM20IR 44585259 IC50 = 315.9 nM T65755 C02XSJ 44585260 IC50 = 31.7 nM T65755 C4WKI8 44585264 IC50 = 1.9 nM T65755 C3UM5R 44585265 IC50 = 5.4 nM T65755 CU0C7J 44585266 IC50 = 162.6 nM T65755 CM9ON1 44585267 IC50 = 2.3 nM T65755 C2T0IE 44585272 IC50 = 16.6 nM T65755 CI6T1Y 44585273 IC50 = 2.1 nM T65755 CKM86B 44585274 IC50 = 151.5 nM T65755 CEIU92 44585332 IC50 = 15.3 nM T65755 C7DS4E 44585337 IC50 = 110 nM T65755 C0H3DC 44585346 IC50 = 112.5 nM T65755 C3ZO2S 44585347 IC50 = 23.9 nM T65755 CC7Q0K 44585348 IC50 = 43.4 nM T65755 C2UA3H 44585349 IC50 = 31.9 nM T65755 C65WDJ 44585350 IC50 = 17.4 nM T65755 CGI7Q1 44589524 EC50 = 120 nM T65755 C02NAI 44589525 EC50 = 93 nM T65755 C9RA0C 44589548 EC50 = 38 nM T65755 CWY59B 44589549 EC50 = 190 nM T65755 C0IAR1 44589552 EC50 = 29 nM T65755 CZVO54 44589735 EC50 = 10000 nM T65755 CZNQ90 44593458 IC50 > 100000 nM T65755 CH2J8R 44598238 IC50 = 1009 nM T65755 CE5W3U 44598288 IC50 = 253 nM T65755 C68BJH 44598289 IC50 = 1010 nM T65755 C9K2WV 44598290 IC50 = 500 nM T65755 CGT51H 44598480 IC50 = 54 nM T65755 CO5YJ8 44598535 IC50 = 205 nM T65755 CO7S9W 44626297 IC50 = 900 nM T65755 C3LIV1 44819032 IC50 = 85 nM T65755 CAQ0C6 44819384 IC50 = 20 nM T65755 C87NFV 44819728 IC50 = 323 nM T65755 CI86ZT 44820090 IC50 = 1480 nM T65755 CXR3J0 45140149 IC50 = 3.4 nM T65755 C42EAO 45140150 IC50 = 39.6 nM T65755 CQ0WZ2 45140151 IC50 = 121.7 nM T65755 CCLE50 45140153 IC50 = 4.2 nM T65755 C4QVP3 45140347 IC50 = 5.6 nM T65755 CR8GN7 45140348 IC50 = 25.7 nM T65755 C6K1JW 45140349 IC50 = 98.4 nM T65755 C82WLQ 45140350 IC50 = 165.3 nM T65755 CR4C9A 45140351 IC50 = 188 nM T65755 C3TIZ2 45263266 IC50 = 26150 nM T65755 CBVG47 45263294 IC50 = 58970 nM T65755 CP7LW4 45263306 IC50 = 25140 nM T65755 C7I5HL 45263307 IC50 = 80250 nM T65755 C72TGV 45265748 IC50 = 98520 nM T65755 C0LKV3 45265776 IC50 = 40010 nM T65755 CC24IR 45276264 IC50 = 5620000 nM T65755 C96ROY 45482635 IC50 > 50000 nM T65755 C02LVF 45485792 IC50 = 17 nM T65755 C1TL8U 45485793 IC50 = 791 nM T65755 CQM78O 45485819 IC50 = 541 nM T65755 CT0PS6 46200966 IC50 = 2.8 nM T65755 CW6YM2 46225959 IC50 = 0.9 nM T65755 CC6FS7 46225960 IC50 = 1.2 nM T65755 CC5VT8 46225961 IC50 = 7 nM T65755 C7CQ1I 46225962 IC50 = 0.95 nM T65755 C7AS6B 46225963 IC50 = 11 nM T65755 CHR7O8 46225964 IC50 = 1 nM T65755 CV8W2O 46225965 IC50 = 2.1 nM T65755 CYTX59 46225966 IC50 = 2 nM T65755 CD1O7V 46225967 IC50 = 6.9 nM T65755 C7LEI9 46225968 IC50 = 7 nM T65755 C8OLF0 46225969 IC50 = 1.2 nM T65755 C95BSV 46225970 IC50 = 3.3 nM T65755 CX2AY0 46226795 IC50 = 40000 nM T65755 CQO2B0 46226895 IC50 = 8 nM T65755 C2P6XR 46229559 IC50 = 108.9 nM T65755 C2PD1Y 46229560 IC50 = 147.7 nM T65755 C8CMV0 46229585 IC50 = 226.1 nM T65755 CH47GM 46229586 IC50 = 212.9 nM T65755 CJIW73 46229683 IC50 = 596.6 nM T65755 C54BRN 46229700 IC50 = 55.4 nM T65755 C5FVI9 46231287 IC50 = 510 nM T65755 C3FE0U 46231288 IC50 = 360 nM T65755 CNQY52 46231327 IC50 = 290 nM T65755 CM4W2T 46231328 IC50 = 300 nM T65755 CS8P3R 46233390 IC50 = 11.3 nM T65755 CN25IK 46844536 IC50 = 8.9 nM T65755 C30YCD 46881260 IC50 = 347000 nM T65755 C48QWG 46884058 IC50 = 215 nM T65755 CVU0D3 46884059 IC50 = 21 nM T65755 C5UMJ3 46884060 IC50 = 26 nM T65755 CQ76JG 46884061 IC50 = 206 nM T65755 C9HMN4 46884114 IC50 = 171 nM T65755 C8V3HK 46884115 IC50 = 141 nM T65755 C8CI2D 46884116 IC50 = 615 nM T65755 C35OPR 46884117 IC50 = 20 nM T65755 CI0W9C 46884118 IC50 = 35 nM T65755 C25DSY 46887918 IC50 = 133 nM T65755 C93CLK 46887919 IC50 = 23600 nM T65755 CY0G9N 46905060 IC50 = 50640 nM T65755 CKCJ01 46906239 IC50 = 50000 nM T65755 C0C3HL 46906265 IC50 = 32000 nM T65755 CL40MY 46906266 IC50 = 82850 nM T65755 C07SUF 46906297 IC50 = 179400 nM T65755 CBC2M7 46907394 IC50 = 19 nM T65755 CLY8Q9 46907395 IC50 < 1 nM T65755 C3ZLJ2 46907396 IC50 = 300 nM T65755 C7YA1I 46907405 IC50 = 2700 nM T65755 CFI74D 46907406 IC50 = 2000 nM T65755 CA4DJ0 46907407 IC50 = 40 nM T65755 C4MN3R 46907408 IC50 > 10000 nM T65755 CY7B1U 46913905 IC50 = 163.6 nM T65755 C42UBP 46913906 IC50 = 208.2 nM T65755 CWA0M8 46916092 IC50 = 7.77 nM T65755 CYN9W5 46916093 IC50 = 1.03 nM T65755 C78XOJ 46916094 IC50 = 104.2 nM T65755 C51QUX 49846125 IC50 = 160 nM T65755 CFZL34 49846205 IC50 = 110 nM T65755 CDI98R 49846207 IC50 = 120 nM T65755 CGL24M 49846275 IC50 = 320 nM T65755 CNM45I 49846277 IC50 = 70 nM T65755 CUC04Q 49846349 IC50 = 70 nM T65755 CJ5C2N 49846418 IC50 = 30 nM T65755 CQ0YP8 49846419 IC50 = 420 nM T65755 C72XMT 49846623 IC50 = 100 nM T65755 CG8E7U 49846694 IC50 = 90 nM T65755 CR8BS4 49846841 IC50 = 310 nM T65755 CLW5T3 49846920 IC50 = 190 nM T65755 C35CDV 49846990 IC50 = 100 nM T65755 CMJE07 49846991 IC50 = 230 nM T65755 C2N1VI 49846994 IC50 = 150 nM T65755 CGYV81 49846995 IC50 = 380 nM T65755 C7DKE3 49847075 IC50 = 480 nM T65755 CJE36W 49847076 IC50 = 210 nM T65755 C0S2JO 49847146 IC50 = 30 nM T65755 C8RWO1 49847147 IC50 = 140 nM T65755 CIU0G4 49847151 IC50 = 100 nM T65755 C58AIU 49847221 IC50 = 380 nM T65755 CP3S8L 49847227 IC50 = 70 nM T65755 CC7Y9U 49850262 IC50 = 9900 nM T65755 C8V3ED 49855395 IC50 = 23 nM T65755 CE7D2J 49855568 IC50 = 630 nM T65755 CFD9P3 49855569 IC50 = 50000 nM T65755 CPGO64 49855588 IC50 = 32 nM T65755 C5LY6T 49855593 IC50 = 6.5 nM T65755 CRFX39 49855594 IC50 = 27 nM T65755 C1AU5N 49855758 IC50 > 32000 nM T65755 CIFK93 49855759 IC50 > 100000 nM T65755 CK48OJ 49855760 IC50 > 10000 nM T65755 CZI3M1 49855761 IC50 > 32000 nM T65755 C9ORU7 49855789 IC50 = 13 nM T65755 C51KYC 49855790 IC50 = 40 nM T65755 CRPZ58 49855949 IC50 > 32000 nM T65755 CTU0K3 49855950 IC50 > 32000 nM T65755 CF85NL 49855951 IC50 > 32000 nM T65755 CF7YS9 49855952 IC50 = 8300 nM T65755 CJU38G 49855953 IC50 = 430 nM T65755 C96HUF 49855976 IC50 = 57 nM T65755 C0N7RV 49856926 IC50 = 12.4 nM T65755 C7ER8Q 49856927 IC50 = 10 nM T65755 C67LXH 49856928 IC50 = 34 nM T65755 C6J4FS 49856929 IC50 = 44 nM T65755 CW20LP 49856930 IC50 = 27 nM T65755 C6POK9 49856931 IC50 = 13 nM T65755 C1JTA8 49856932 IC50 = 14 nM T65755 CG2A8T 49857123 IC50 = 34 nM T65755 CHG64R 49857124 IC50 = 16 nM T65755 C36AWV 49857125 IC50 = 30 nM T65755 CUK9R8 49857126 IC50 = 15 nM T65755 C2BL6I 49857127 IC50 = 20 nM T65755 C5FTK3 49857128 IC50 = 22 nM T65755 C46IQN 49857313 IC50 = 16 nM T65755 CE6B3A 49857314 IC50 = 16 nM T65755 CX0N2J 49857315 IC50 = 14 nM T65755 CS40UV 49857316 IC50 = 9 nM T65755 C6YPD7 49864403 IC50 = 85000 nM T65755 CD5J7W 50898619 IC50 = 13 nM T65755 C4P8YF 50898980 IC50 = 9400 nM T65755 C5Z6GI 50898981 IC50 = 61100 nM T65755 CP30HY 50898982 IC50 = 87500 nM T65755 CA7BW0 50898983 IC50 = 58100 nM T65755 COA5W3 51051073 IC50 = 26 nM T65755 C3AQ4J 51353583 IC50 = 62 nM T65755 CGY6F0 51353584 IC50 = 183 nM T65755 CB30WO 51353585 IC50 = 114 nM T65755 C1TR7X 51356437 IC50 = 131 nM T65755 CBF46X 51356438 IC50 = 955 nM T65755 C1KTN8 51356439 IC50 = 187 nM T65755 CA6YL2 51356710 IC50 = 119 nM T65755 CR16LM 51356712 IC50 = 27 nM T65755 CY8A4B 51356714 IC50 = 196 nM T65755 CIZ51T 51356715 IC50 = 136 nM T65755 CRZ95L 51356716 IC50 = 56 nM T65755 C3AI5C 51356989 IC50 = 237 nM T65755 CTUC09 51356990 IC50 = 232 nM T65755 CA40OC 51356991 IC50 = 207 nM T65755 CC7O2B 51356993 IC50 = 34 nM T65755 C81BOJ 51356994 IC50 = 1 nM T65755 C7M6DH 51356995 IC50 = 165 nM T65755 C2HD5S 51357269 IC50 = 134 nM T65755 CV76KB 51357270 IC50 = 73 nM T65755 CL56AW 51357271 IC50 = 323 nM T65755 CN3M2Z 51357272 IC50 = 110 nM T65755 C4L9AP 51357273 IC50 = 114 nM T65755 CJD70E 51357274 IC50 = 300 nM T65755 CV4L0J 51357275 IC50 = 56 nM T65755 C1YZU0 51357550 IC50 = 149 nM T65755 CHTP31 51357551 IC50 = 228 nM T65755 C7L9JO 51357552 IC50 = 67 nM T65755 CD0M2K 51357553 IC50 = 219 nM T65755 CP37JA 51357554 IC50 = 130 nM T65755 C4K2WT 51357555 IC50 = 168 nM T65755 CV5DF8 51357823 IC50 = 485 nM T65755 C1WKN9 51357824 IC50 = 81 nM T65755 CDUN82 51357825 IC50 = 286 nM T65755 CUY3W2 52918057 IC50 = 840 nM T65755 CKZ8U0 52918058 IC50 = 260 nM T65755 C20SMD 52918059 IC50 = 100 nM T65755 C4RM1H 52918060 IC50 = 90 nM T65755 CWRD28 52918061 IC50 = 540 nM T65755 CCBZ05 52941022 IC50 = 42 nM T65755 CTK72Z 52942121 IC50 = 122 nM T65755 CYD47V 52942292 IC50 = 30 nM T65755 CT2FC9 52943493 IC50 = 50 nM T65755 C9VG2Q 52945663 IC50 = 64 nM T65755 C7QRS9 52945665 IC50 = 433 nM T65755 CY2U3W 52945750 IC50 = 12 nM T65755 C94LPE 52945855 IC50 = 45 nM T65755 C2F3LB 52947746 IC50 = 95 nM T65755 C10YJQ 52949337 IC50 = 123 nM T65755 CR4P8B 52951037 IC50 = 5840 nM T65755 CHX3K6 52951172 IC50 = 538 nM T65755 CYU0R2 52951254 IC50 = 65 nM T65755 C78BHS 52951255 IC50 = 128 nM T65755 C08BSF 52951359 IC50 = 214 nM T65755 CNC9V0 52951361 IC50 = 108 nM T65755 CSX0H2 52951363 IC50 = 73 nM T65755 C2IXJ1 52951365 IC50 = 71 nM T65755 CSB58V 52951464 IC50 = 447 nM T65755 CZ9FU4 52951465 IC50 = 297 nM T65755 CG87BZ 52952415 IC50 > 50000 nM T65755 C2J8VC 52952416 IC50 > 50000 nM T65755 CA4O8L 52952417 IC50 = 24000 nM T65755 C0AMH6 52952418 IC50 = 29000 nM T65755 C6DAB7 52952491 IC50 = 58 nM T65755 CVBE93 53258999 IC50 = 120 nM T65755 CR2SH5 53317649 EC50 = 2650 nM T65755 CLRT20 53317827 IC50 = 44 nM T65755 CM3V9P 53323775 EC50 = 280 nM T65755 CWPI96 53325741 IC50 = 420 nM T65755 C9JK4A 53326649 IC50 = 7.6 nM T65755 CATU50 53357596 IC50 = 358 nM T65755 C5AQC7 53357597 IC50 = 1320 nM T65755 CN0QR2 53357716 IC50 = 889 nM T65755 C9WL1R 53387509 IC50 = 52 nM T65755 C1OT3A 53464575 IC50 > 1000 nM T65755 C9U7GF 53464577 IC50 = 29.5 nM T65755 C4EYP7 53464578 IC50 = 6.8 nM T65755 C0WNH9 53464579 IC50 = 16.8 nM T65755 C4MQ3U 53464638 IC50 = 9.7 nM T65755 CJ53ZV 53464639 IC50 = 32.1 nM T65755 CX4Z0I 53464640 IC50 = 757.6 nM T65755 CLNR63 53464641 IC50 = 186.5 nM T65755 CLCK01 53464704 IC50 > 1000 nM T65755 C5VRU2 53464705 IC50 = 254 nM T65755 CD07PL 53464707 IC50 > 1000 nM T65755 CXQN21 53464764 IC50 = 275.2 nM T65755 CN9RH2 53464770 IC50 = 12.6 nM T65755 C0ZK7I 54576529 IC50 = 28.9 nM T65755 CTP2S1 54576530 IC50 = 24.6 nM T65755 CS8HY5 54576744 IC50 = 22.2 nM T65755 C5H9SW 54584126 IC50 = 1390 nM T65755 CU3H0Y 54753628 IC50 = 350 nM T65755 CVP16C 54753629 IC50 = 32000 nM T65755 CO87WU 54770222 IC50 = 426.3 nM T65755 CC1IU2 54770436 IC50 = 209.9 nM T65755 CX9C5K 54770437 IC50 = 523.2 nM T65755 C3IJ0Z 54770438 IC50 = 128.2 nM T65755 CMZ6I8 54770439 IC50 = 39 nM T65755 CGB9A6 54770440 IC50 = 711.6 nM T65755 C7PS9X 54770441 IC50 = 425.5 nM T65755 CQ1EX7 54770442 IC50 = 23.7 nM T65755 C9IJ0S 54770657 IC50 = 111.7 nM T65755 CBT20G 56657793 IC50 = 235 nM T65755 C0S5IE 56657800 IC50 = 34 nM T65755 C5NV0G 56657801 IC50 = 13 nM T65755 CIU42S 56657802 IC50 = 0.2 nM T65755 CAXH26 56657895 IC50 = 61 nM T65755 C0TB5E 56657896 IC50 = 0.3 nM T65755 CV18MG 56657897 IC50 = 1 nM T65755 CA70SC 56658395 IC50 = 184000 nM T65755 CP8RN3 56659683 IC50 = 1230 nM T65755 CIC29M 56661386 IC50 = 110 nM T65755 C61RBI 56661387 IC50 = 73 nM T65755 C3B5AL 56661409 IC50 = 450 nM T65755 CGO3P6 56661410 IC50 = 1 nM T65755 CVP3U1 56661411 IC50 = 18 nM T65755 CW15JN 56661412 IC50 = 848 nM T65755 CM8V0L 56661413 IC50 = 39 nM T65755 C3L6YS 56664683 IC50 = 0.005 ug.mL-1 T65755 CNU92J 56664684 IC50 = 0.01 ug.mL-1 T65755 CL85AP 56664859 IC50 = 700 nM T65755 CU3WQ7 56668109 IC50 = 0.7 ug.mL-1 T65755 C4GY3I 56668199 IC50 = 1 nM T65755 CDQG86 56668203 IC50 = 0.2 nM T65755 CMV01S 56668204 IC50 = 1.3 nM T65755 CQV53G 56668278 IC50 = 60 nM T65755 C1JSP2 56668279 IC50 = 85 nM T65755 CE8B4S 56668280 IC50 = 0.4 nM T65755 C6WVO2 56668281 IC50 = 180 nM T65755 C9AZ8J 56668283 IC50 = 30 nM T65755 C4ORP6 56668284 IC50 = 15 nM T65755 CK1AG3 56668788 IC50 = 15000 nM T65755 CBHX35 56671569 IC50 = 2 ug.mL-1 T65755 CO4QU3 56671735 IC50 = 85 nM T65755 C7UFS3 56671736 IC50 = 3 nM T65755 CPE64C 56671747 IC50 = 1450 nM T65755 CU1IN2 56671748 IC50 = 144 nM T65755 C05XIJ 56671749 IC50 < 0.1 nM T65755 C6CQ7B 56671750 IC50 = 2000 nM T65755 CT2LE0 56671751 IC50 = 110 nM T65755 CV35BF 56675013 IC50 = 5 ug.mL-1 T65755 CWMU10 56675096 IC50 = 444 nM T65755 CXR38G 56675097 IC50 = 67 nM T65755 CH2NY9 56675158 IC50 = 6 nM T65755 CGAI64 56675159 IC50 = 5 nM T65755 C0IJ5Z 56678453 IC50 = 74 nM T65755 CE2G8K 56678454 IC50 = 2 nM T65755 CM6XD8 56678455 IC50 = 326 nM T65755 CY4AQ1 56678470 IC50 = 0.2 nM T65755 C76PCA 56678471 IC50 = 7 nM T65755 CTC08Y 56678472 IC50 = 282 nM T65755 CZ4HY1 56678965 IC50 = 73000 nM T65755 C79RJG 56679976 IC50 = 18 nM T65755 C5Z0PH 56681671 IC50 = 1 ug.mL-1 T65755 C6YUD2 56681816 IC50 = 85 nM T65755 C8NS0H 56683541 IC50 = 3.3 nM T65755 C2ML5S 56837168 IC50 = 935 nM T65755 C78VPM 56928522 IC50 = 213 nM T65755 CCW89V 56932477 IC50 = 117 nM T65755 CTS0R7 56932478 IC50 = 443 nM T65755 C41ZBJ 56951446 IC50 = 14000 nM T65755 C1R7HZ 56951447 IC50 = 49000 nM T65755 C4DZ0B 57336556 IC50 > 50000 nM T65755 CN9W2G 57336559 IC50 > 50000 nM T65755 C10DMC 57336560 IC50 > 50000 nM T65755 CU6B5H 57336562 IC50 = 42000 nM T65755 C8O0CH 57336568 IC50 = 45000 nM T65755 C5CN3K 57336569 IC50 > 50000 nM T65755 C0BT1I 57336572 IC50 > 50000 nM T65755 CNHJ96 57394371 IC50 = 537 nM T65755 CYSH27 57396190 IC50 = 317 nM T65755 C5CRJ1 57412107 IC50 = 108 nM T65755 COG4Q8 57412108 IC50 = 113 nM T65755 CR07DZ 57413556 IC50 = 170.9 nM T65755 CAH3K1 57413557 IC50 > 1000 nM T65755 C68ZKL 57413558 IC50 = 407.5 nM T65755 CWYI96 57658333 IC50 = 1760 nM T65755 CND60S 58147877 IC50 = 174 nM T65755 C2A5FR 58147881 IC50 = 667 nM T65755 C3TBY4 58147895 IC50 = 645 nM T65755 CV87YQ 58147896 IC50 = 59 nM T65755 C4V7FY 58191950 IC50 = 4240 nM T65755 CPCA29 58191961 IC50 = 34 nM T65755 C7HF1L 58191965 IC50 = 200 nM T65755 CR4BX0 58191982 IC50 > 15800 nM T65755 C8V1NK 58191988 IC50 > 15800 nM T65755 C8LWY9 58191997 IC50 = 2460 nM T65755 C3IQ9B 58191999 IC50 = 380 nM T65755 CQB69R 58192003 IC50 > 15800 nM T65755 C42FDY 60163732 IC50 = 6700 nM T65755 CXRF43 70681934 IC50 = 1890 nM T65755 CLK09M 70681935 IC50 = 3650 nM T65755 CX5VN1 70681936 IC50 = 3270 nM T65755 CS30XY 70684051 IC50 = 3590 nM T65755 C9OT4C 70684052 IC50 = 3480 nM T65755 C6A8OR 70684387 IC50 = 53 nM T65755 C4M2OY 70686190 IC50 = 6020 nM T65755 CQE6H8 70686191 IC50 = 3020 nM T65755 C8KS2X 70690332 IC50 = 3190 nM T65755 C29RZD 70690333 IC50 = 2030 nM T65755 CM9C6X 70690334 IC50 = 1210 nM T65755 CI4WH5 70690843 IC50 > 100000 nM T65755 CW45VZ 70692855 IC50 = 111 nM T65755 CO1MU8 70694542 IC50 = 3010 nM T65755 C9D4UF 70694543 IC50 = 1860 nM T65755 CA0CP1 70694544 IC50 = 560 nM T65755 C5D0JG 70694885 IC50 = 42 nM T65755 CBFK85 70694886 IC50 = 60 nM T65755 C6HI8Q 70696598 IC50 = 4090 nM T65755 CBCF23 70696599 IC50 = 1090 nM T65755 CL5J4X 70696942 IC50 = 153 nM T65755 C3J9QZ 71453454 IC50 = 250 nM T65755 CIU86S 71453462 IC50 = 18000 nM T65755 C87VDX 71455164 IC50 > 100000 nM T65755 C57ATO 71455172 IC50 = 1000 nM T65755 CH7X0R 71455807 IC50 = 456 nM T65755 C7RLK3 71455808 IC50 = 344 nM T65755 C6B2HJ 71456958 IC50 = 60 nM T65755 CYIW96 71456964 IC50 > 100000 nM T65755 CHS8I5 71456965 IC50 > 100000 nM T65755 C4V7EN 71456966 IC50 > 10000 nM T65755 C76SGF 71457594 IC50 = 1940 nM T65755 CM9A3I 71458827 IC50 = 210 nM T65755 C3U2YL 71458828 IC50 > 10000 nM T65755 CHO52U 71459490 IC50 = 349 nM T65755 CP58UV 71460639 IC50 > 10000 nM T65755 CR43ZN 71462354 IC50 > 100000 nM T65755 CB1N8K 71462355 IC50 > 10000 nM T65755 CZ1S7V 71506894 IC50 = 100 nM T65755 C01XHF 71510730 IC50 = 158 nM T65755 C09YSR 71510731 IC50 = 123 nM T65755 CV5R8E 71520424 IC50 = 1700 nM T65755 C38UCW 71520532 IC50 = 1660 nM T65755 CPV4L5 71520533 IC50 = 1430 nM T65755 C4NO1T 71520534 IC50 = 5730 nM T65755 CXR70T 71520535 IC50 = 900 nM T65755 CFQ2N9 71520536 IC50 = 1070 nM T65755 CS6NP3 71520537 IC50 = 2050 nM T65755 C29SEZ 71520538 IC50 = 1320 nM T65755 C3A6EJ 71520539 IC50 = 8860 nM T65755 CGLW63 71520625 IC50 = 7630 nM T65755 CMP8E3 71520626 IC50 = 4640 nM T65755 C2NG6H 71520627 IC50 = 1260 nM T65755 C3K9FG 71520628 IC50 = 2000 nM T65755 C3DC4O 71520629 IC50 = 1950 nM T65755 CI0H5Y 71520630 IC50 = 600 nM T65755 C0LWJ6 71520631 IC50 = 1130 nM T65755 CL7RD9 71520632 IC50 = 4210 nM T65755 CNT81Q 71520633 IC50 = 15400 nM T65755 CO28HI 71520716 IC50 = 880 nM T65755 CVA5Q7 71520717 IC50 = 320 nM T65755 CGL95K 71521451 IC50 = 15200 nM T65755 C4FLX8 71521452 IC50 > 100000 nM T65755 CIY52O 71521453 IC50 = 4950 nM T65755 CM6FL5 71521531 IC50 = 34000 nM T65755 CP78KS 71521532 IC50 = 43900 nM T65755 C98QLB 71521701 IC50 > 100000 nM T65755 C93DWO 71521702 IC50 > 100000 nM T65755 C7SN9R 71527845 IC50 = 2910 nM T65755 C6S5JQ 71527847 IC50 = 1080 nM T65755 CVOF76 71527974 IC50 = 620 nM T65755 C4XEO5 71527975 IC50 = 380 nM T65755 C2FVD0 71527976 IC50 = 160 nM T65755 C16AHW 71527977 IC50 = 180 nM T65755 C2VA7F 71528083 IC50 = 430 nM T65755 C7KB2M 71528084 IC50 = 180 nM T65755 C3E9XO 71528085 IC50 = 140 nM T65755 C0E1YJ 71528086 IC50 = 320 nM T65755 CXI8D3 71528200 IC50 = 430 nM T65755 CQ7RA2 71528201 IC50 = 1170 nM T65755 CTJF80 71528202 IC50 = 800 nM T65755 C6O8UK 71528203 IC50 = 730 nM T65755 CMR1K9 71528318 IC50 = 710 nM T65755 CE0K6S 71535880 IC50 = 610.5 nM T65755 CV6Q3H 71535881 IC50 = 2090 nM T65755 CKC89T 71535884 IC50 = 490 nM T65755 C5Z6IU 71536146 IC50 = 170 nM T65755 CK1PT4 71536148 IC50 = 570 nM T65755 CRIQ61 71536691 IC50 = 1120 nM T65755 CP5N7Z 71536967 IC50 = 1060 nM T65755 CA19SE 71536968 IC50 = 1470 nM T65755 CJDS45 71538210 IC50 = 200 nM T65755 CBV1C3 71625213 IC50 = 250 nM T65755 C6YAV2 71625223 IC50 = 155.4 nM T65755 CLW8K3 71625224 IC50 = 120.7 nM T65755 C53BQN 71625225 IC50 = 64.65 nM T65755 C4U1LY 71625326 IC50 = 214 nM T65755 CCQ0U1 71625341 IC50 = 212.3 nM T65755 COZX76 71625342 IC50 = 144.5 nM T65755 C1PAI9 71625343 IC50 = 112.2 nM T65755 CD09SV 71625344 IC50 = 56.2 nM T65755 C6V7JB 71625441 IC50 = 298 nM T65755 CHR9E5 71625445 IC50 = 140 nM T65755 C02PZB 71625559 IC50 = 164 nM T65755 CW87PT 71625562 IC50 = 157 nM T65755 CPJ4V7 71680913 IC50 = 6700 nM T65755 CWOJ34 71698768 IC50 = 78 nM T65755 CMV8P7 71698769 IC50 = 204 nM T65755 CPH53O 71698854 IC50 = 99 nM T65755 CI2L0Q 71698938 IC50 = 103 nM T65755 CNF6I3 71698939 IC50 = 91 nM T65755 C7IU1F 71699034 IC50 = 527 nM T65755 CV0Y5P 71699035 IC50 = 136 nM T65755 C5T2MQ 71699036 IC50 = 137 nM T65755 C9T0HW 71699037 IC50 = 258 nM T65755 CIY84O 71699121 IC50 = 540 nM T65755 C31RLA 71712310 IC50 = 557 nM T65755 CJ6NY4 71714525 IC50 = 458 nM T65755 CKX92J 71714526 IC50 = 2910 nM T65755 CV4A1N 71714527 IC50 = 9190 nM T65755 CO2B0D 71714528 IC50 = 11630 nM T65755 CGN39Q 71714529 IC50 = 3790 nM T65755 C39WMS 71714530 IC50 = 1350 nM T65755 CT5ZG4 71714531 IC50 = 989 nM T65755 CU0E8S 71714532 IC50 = 1080 nM T65755 C7SIB5 71717929 IC50 = 2.2 nM T65755 CIR56T 71721558 IC50 > 100000 nM T65755 CCD18W 71721946 IC50 > 100000 nM T65755 C6U9VB 71769925 IC50 = 130 nM T65755 CIRH21 71769926 IC50 = 170 nM T65755 C26HDR 71769927 IC50 = 180 nM T65755 C5RXY7 71769928 IC50 = 540 nM T65755 CT1RZ2 71770054 IC50 = 3170 nM T65755 C28JCL 71770055 IC50 = 2650 nM T65755 CEL21O 71770056 IC50 = 2550 nM T65755 CTPJ18 71770057 IC50 = 170 nM T65755 C1TSQ4 71770058 IC50 > 2550 nM T65755 CVU1W6 71770059 IC50 = 1870 nM T65755 CHK58Q 71770060 IC50 = 1480 nM T65755 CG3X4E 71770191 IC50 = 2540 nM T65755 CVO12E 71770192 IC50 = 2120 nM T65755 CJ87KH 71770193 IC50 = 1310 nM T65755 C8J7IV 71770194 IC50 = 1250 nM T65755 C4TF1J 71770195 IC50 = 1610 nM T65755 C7L4DU 71770196 IC50 > 2390 nM T65755 CT0ZN2 71770317 IC50 > 2170 nM T65755 CW4FB0 71770318 IC50 > 2550 nM T65755 CJ7BK6 71770319 IC50 = 89 nM T65755 C4X8RV 71770320 IC50 = 1210 nM T65755 CN5D6Z 71770321 IC50 = 1710 nM T65755 C9K1YU 71770322 IC50 > 2070 nM T65755 CZ2H9B 71770436 IC50 = 1660 nM T65755 CI0T4S 71770437 IC50 > 2020 nM T65755 CJ9K8V 71770438 IC50 > 1960 nM T65755 C13MPI 71770439 IC50 = 2310 nM T65755 CMI5D3 71770440 IC50 = 1590 nM T65755 CMTU70 71770441 IC50 > 2690 nM T65755 CAU01F 71770557 IC50 > 2690 nM T65755 C36OTC 71770558 IC50 = 3490 nM T65755 C5ICX8 71770559 IC50 = 2280 nM T65755 C2PNQ0 71770560 IC50 = 400 nM T65755 CD98TG 71770561 IC50 = 2360 nM T65755 C5K4ZC 71770562 IC50 = 840 nM T65755 CB6D2C 71770683 IC50 > 2220 nM T65755 CY9NF1 71770684 IC50 = 1570 nM T65755 CB9L8Z 72204662 IC50 = 160 nM T65755 CT7M6G 72204663 IC50 = 340 nM T65755 C1VG8U 72204664 IC50 = 180 nM T65755 CC0XI1 72204665 IC50 = 600 nM T65755 C4MW3U 72204666 IC50 = 380 nM T65755 C98VDM 72204667 IC50 = 320 nM T65755 CU30CD 72205221 IC50 = 310 nM T65755 C90FMR 72205411 IC50 = 120 nM T65755 C4WU0F 72543937 IC50 = 234 nM T65755 CP64JM 72543939 IC50 = 186 nM T65755 CZ6TC4 72543940 IC50 = 304 nM T65755 CM1NY3 72543941 IC50 = 410 nM T65755 CN23FO 72544176 IC50 = 210 nM T65755 CHA93V 72544177 IC50 = 130 nM T65755 CENG73 72544178 IC50 = 216 nM T65755 CQF14E 72544179 IC50 = 187 nM T65755 CCGD47 72547524 IC50 = 198 nM T65755 CUHA54 72547525 IC50 = 172 nM T65755 C6AN1B 72547526 IC50 = 206 nM T65755 CU5XH0 72696071 IC50 = 15100 nM T65755 C1F7OV 72696072 IC50 = 64500 nM T65755 CN4AP3 72696073 IC50 = 118000 nM T65755 C46LKB 72696074 IC50 = 16400 nM T65755 C27FNY 72696075 IC50 = 11600 nM T65755 CU8D1K 72696076 IC50 = 66600 nM T65755 CJR3Z7 72696203 IC50 = 71400 nM T65755 CV9F8G 72696204 IC50 = 7430 nM T65755 CO26MJ 72697863 IC50 = 12500 nM T65755 C4S3HG 72697864 IC50 = 43000 nM T65755 CC7UN2 72697865 IC50 = 10800 nM T65755 CXM8W9 72697866 IC50 = 8430 nM T65755 CV3IC2 72697867 IC50 = 3940 nM T65755 CU8W9S 72697868 IC50 = 9470 nM T65755 CGKQ31 72697869 IC50 = 10500 nM T65755 CKP92S 72698003 IC50 = 67800 nM T65755 CA4W8H 72698004 IC50 = 11500 nM T65755 CCBU94 72698005 IC50 = 49600 nM T65755 CZK0R3 72698006 IC50 = 10300 nM T65755 CEC2O3 72698007 IC50 = 8950 nM T65755 C5JNM9 72698008 IC50 = 12800 nM T65755 CFN42K 72698149 IC50 = 73700 nM T65755 C7TFD9 72698150 IC50 = 2820 nM T65755 C1V6HS 72698151 IC50 = 7800 nM T65755 CI5FX8 72698152 IC50 = 24200 nM T65755 C5YO3P 73055009 IC50 = 380 nM T65755 C8A3UJ 73055010 IC50 = 490 nM T65755 CW93JP 73055011 IC50 = 610 nM T65755 C7KU6R 73345517 IC50 = 110 nM T65755 C5P3KB 73347046 IC50 = 7 nM T65755 C6VB1L 73348547 IC50 = 15 nM T65755 CO1V3X 73349613 IC50 = 49300 nM T65755 CN1P0H 73349614 IC50 = 15400 nM T65755 C8NEH3 73350138 IC50 = 74 nM T65755 C1AHE8 73351618 IC50 = 1 nM T65755 C03EUJ 73353105 IC50 < 0.1 nM T65755 C0UQO1 73353605 IC50 = 360 nM T65755 C2O5BM 73354620 IC50 = 0.4 nM T65755 CB8H7V 73356177 IC50 = 0.2 nM T65755 C0D3VA 73504745 IC50 = 5370 nM T65755 C4HMN1 73504960 IC50 = 1210 nM T65755 C6XLM5 73504962 IC50 = 1260 nM T65755 CC0VY1 73505169 IC50 = 3230 nM T65755 CW6K3M 73505171 IC50 = 1560 nM T65755 CXR28I 73505591 IC50 = 3020 nM T65755 CWM70R 73505592 IC50 = 1310 nM T65755 CNC6Q5 73505594 IC50 = 670 nM T65755 CGV9D2 73774761 IC50 > 5000 nM T65755 C9V0AS 73774762 IC50 = 917.4 nM T65755 C81PLN 73774763 IC50 = 439.7 nM T65755 CJ1DA8 73774764 IC50 = 369.8 nM T65755 CQ3K6G 73776326 IC50 = 10.5 nM T65755 CC4L0G 73776327 IC50 = 23.2 nM T65755 C2YJ6R 73776329 IC50 = 636.9 nM T65755 CKAC13 73776470 IC50 = 1703.4 nM T65755 CHX1Y9 73776471 IC50 > 5000 nM T65755 CZB6G7 73776472 IC50 = 5.6 nM T65755 CP69AM 73776473 IC50 = 147.9 nM T65755 C20KBV 73776474 IC50 = 50.4 nM T65755 C0R1SH 73776612 IC50 = 186.5 nM T65755 CVJ4P2 73776613 IC50 = 209.8 nM T65755 CSRE84 73776614 IC50 = 6.7 nM T65755 C10RIN 73776615 IC50 = 20.4 nM T65755 C01FVX 73776616 IC50 = 4.8 nM T65755 C24SLB 73776752 IC50 = 130.3 nM T65755 CC7Z8S 73776753 IC50 = 977.8 nM T65755 CO9R6K 73776897 IC50 = 20.8 nM T65755 CG5D6N 73776898 IC50 = 673.69 nM T65755 CO1E9I 73776899 IC50 = 1043.1 nM T65755 C3UC9H 73891099 IC50 = 9800 nM T65755 CE4MH5 74225266 IC50 = 29800 nM T65755 CWK18T 74226538 IC50 = 19180 nM T65755 CT8D5F 78319205 IC50 = 1370 nM T65755 CB3A0C 78319206 IC50 = 940 nM T65755 CL8HI6 78319207 IC50 = 730 nM T65755 C3IFJ0 78319208 IC50 = 570 nM T65755 C6M9PL 86765212 IC50 = 100 nM T65755 C5U8HL 87258278 IC50 = 150 nM T65755 CBXI21 87258279 IC50 = 85 nM T65755 C5JIT0 87618609 IC50 = 510 nM T65755 CRQO37 88005144 IC50 = 200 nM T65755 C63XNB 89001816 IC50 = 360 nM T65755 CIYO41 89001875 IC50 = 50 nM T65755 CB0S2E 89001876 IC50 = 300 nM T65755 CBE4A5 89001934 IC50 > 10000 nM T65755 C3GE4J 89001938 IC50 = 570 nM T65755 CLYB95 89471379 IC50 = 31 nM T65755 C62GSL 90654859 IC50 = 157.8 nM T65755 C3H6SG 90656558 IC50 > 100000 nM T65755 CFE10C 90656560 IC50 > 100000 nM T65755 CD4L8R 90656562 IC50 > 100000 nM T65755 CEST81 90656564 IC50 > 100000 nM T65755 C7J0CO 90656566 IC50 > 100000 nM T65755 CE9Y4D 90656568 IC50 > 100000 nM T65755 CZVG63 90656570 IC50 > 100000 nM T65755 CT0QG6 90656572 IC50 > 100000 nM T65755 CFPR48 90656574 IC50 > 100000 nM T65755 CDF06N 90656576 IC50 > 100000 nM T65755 CQ3R1A 90656578 IC50 > 100000 nM T65755 CWV0Z9 90656580 IC50 > 100000 nM T65755 CGX01J 90656582 IC50 > 100000 nM T65755 C6M1VH 90656584 IC50 > 100000 nM T65755 C1GUD2 90656586 IC50 > 100000 nM T65755 C5KWT1 90656588 IC50 > 100000 nM T65755 CS7PZ6 90656590 IC50 > 100000 nM T65755 CGF9P3 90656592 IC50 > 100000 nM T65755 CM46JO 90656594 IC50 > 100000 nM T65755 CXL84V 90656596 IC50 > 100000 nM T65755 C7EIO6 90656598 IC50 > 100000 nM T65755 CRH7F2 90656600 IC50 > 100000 nM T65755 CKW64G 90656602 IC50 > 100000 nM T65755 C4CU3D 90656604 IC50 > 100000 nM T65755 C15WHB 90656724 IC50 = 480 nM T65755 CER17P 90670108 IC50 = 530.7 nM T65755 C5UOG7 90670109 IC50 = 600.1 nM T65755 CPX56E 90670110 IC50 = 96.6 nM T65755 CG92XP 90670111 IC50 = 255.1 nM T65755 C0DP2G 90670112 IC50 = 97.6 nM T65755 CG17QJ 90670113 IC50 = 84.3 nM T65755 CIY19C 90670114 IC50 = 52.3 nM T65755 CH7CY0 90670115 IC50 = 198.5 nM T65755 CK3CW6 90670116 IC50 = 148 nM T65755 CJC56B 90670117 IC50 = 447.6 nM T65755 CX28KF 90675408 IC50 = 5820 nM T65755 C49ISO 90675409 IC50 = 2960 nM T65755 CSI27E 90675410 IC50 = 2810 nM T65755 CU9C3N 90675411 IC50 = 4910 nM T65755 CUFD65 90675412 IC50 = 9040 nM T65755 C8OBM4 90675413 IC50 = 66520 nM T65755 CUEI29 90675414 IC50 = 22160 nM T65755 C8AF7R 90675415 IC50 > 200000 nM T65755 CSE5X4 90675416 IC50 = 49300 nM T65755 C9MQV8 90675417 IC50 > 200000 nM T65755 CGMY72 90675418 IC50 = 15600 nM T65755 CXD53P 90675419 IC50 = 24010 nM T65755 C7FTE8 90675420 IC50 > 200000 nM T65755 CIJ4B5 90675421 IC50 > 200000 nM T65755 CRCD95 90675422 IC50 = 31320 nM T65755 CM38TL 90675423 IC50 > 200000 nM T65755 C3H9WM 90675424 IC50 > 200000 nM T65755 CL45KD 90675425 IC50 = 164610 nM T65755 CKPU38 90675426 IC50 = 58240 nM T65755 CRL5J6 90675427 IC50 = 29500 nM T65755 C7JG1Z 90675428 IC50 = 71020 nM T65755 CX3A4C 90675429 IC50 = 56710 nM T65755 CTYW06 90675430 IC50 = 124670 nM T65755 CG9MO0 90676506 IC50 = 510 nM T65755 C03AGY 90676507 IC50 = 230 nM T65755 CM2HG7 90676508 IC50 = 500 nM T65755 CZD65S 90676509 IC50 = 560 nM T65755 CMB30T 90676510 IC50 = 240 nM T65755 CAJI89 90676511 IC50 = 600 nM T65755 CVBA53 90676512 IC50 = 850 nM T65755 C03XSK 91884577 IC50 = 6000 nM T65755 CT7Z8F 102514716 IC50 = 370 nM T65755 C1FL7E 118708140 IC50 = 6.4 nM T65755 CX89LF 118712700 IC50 = 3.3 nM T65755 CG27EL 118712701 IC50 = 2.8 nM T65755 C4OMG6 118712702 IC50 = 3.4 nM T65755 C3M2WV 118712703 IC50 = 7.9 nM T65755 CP5NL9 118712704 IC50 = 7.3 nM T65755 CRN2P8 118712705 IC50 = 47.4 nM T65755 CN89TK 118712706 IC50 = 29.6 nM T65755 CFJZ58 118712707 IC50 = 9.2 nM T65755 C4R3LE 118712708 IC50 = 6.6 nM T65755 CT3Y5U 118712709 IC50 = 5.7 nM T65755 C9V0RX 118712710 IC50 = 43.9 nM T65755 C6YUM5 118712711 IC50 = 771.8 nM T65755 CIYD57 118712713 IC50 = 7.5 nM T65755 C0HO7R 118712965 IC50 = 34000 nM T65755 C8JY2S 118712967 IC50 = 30000 nM T65755 CY6IQ4 118712968 IC50 > 50000 nM T65755 C78MZY 118712969 IC50 = 42000 nM T65755 C0M3XQ 118712970 IC50 > 50000 nM T65755 CMF83S 118712971 IC50 = 48000 nM T65755 C5V6PJ 118720516 IC50 = 886.4 nM T65755 CUMG39 118720517 IC50 = 861.5 nM T65755 C9UP4R 118720518 IC50 = 447.7 nM T65755 CC27SV 118720519 IC50 = 464.5 nM T65755 CD2XP4 118720520 IC50 = 498.6 nM T65755 C1YQ7N 118720521 IC50 = 692.4 nM T65755 CSC47W 118720522 IC50 = 191.2 nM T65755 C8I5OJ 118720523 IC50 = 218.7 nM T65755 CEHQ26 118720524 IC50 = 81.9 nM T65755 C4COD1 118720525 IC50 = 357.9 nM T65755 CIM70O 118720526 IC50 = 258.9 nM T65755 CEV3I6 118720527 IC50 = 779 nM T65755 CEC91V 118720528 IC50 = 67.4 nM T65755 CUI51W 118720529 IC50 = 38.5 nM T65755 CCGH73 118720703 IC50 = 18600 nM T65755 CN2SA5 118734641 IC50 = 251 nM T65755 CF6J5Q 118734642 IC50 = 152 nM T65755 CMHF86 118734643 IC50 = 87 nM T65755 CUE83V 118734644 IC50 = 848 nM T65755 C67IDL 118734645 IC50 = 310 nM T65755 CFD82L 118734646 IC50 = 355 nM T65755 C26ZJS 118734647 IC50 = 159 nM T65755 CM5A9U 118734648 IC50 = 402 nM T65755 C7HP6N 118734649 IC50 = 293 nM T65755 CVIN49 118734650 IC50 = 334 nM T65755 CG8Y5X 118737948 IC50 = 460 nM T65755 C1P2YC 118737949 IC50 = 3940 nM T65755 CXER98 118737950 IC50 = 380 nM T65755 CS71XH 122195525 IC50 = 645 nM T65755 C3AY9G 122195526 IC50 = 121 nM T65755 C2ZY0G 122195527 IC50 = 17 nM T65755 CFYL41 122195528 IC50 = 5.4 nM T65755 CS0NH6 122195529 IC50 = 531 nM T65755 C9JPK0 122195530 IC50 = 97 nM T65755 CEJB32 122195531 IC50 = 15 nM T65755 CFZ54V 122195532 IC50 = 4.5 nM T65755 CNOC04 122195533 IC50 = 215 nM T65755 CV2ZX8 122195534 IC50 = 86 nM T65755 C1LZB0 122195535 IC50 = 14 nM T65755 CW1HK5 122195536 IC50 = 2.8 nM T65755 C2K4OG 122195537 IC50 = 348 nM T65755 CH79VD 122195538 IC50 = 57 nM T65755 CZ9P8V 122195539 IC50 = 21 nM T65755 CR6Q2V 122195540 IC50 = 8.4 nM T65755 CZE35C 122648343 IC50 = 3.4 nM T65755 C54RNT 122648367 IC50 = 3.2 nM T65755 C1UVI7 122648600 IC50 = 6.1 nM T65755 CMX59K 122648648 IC50 = 3.3 nM T65755 CVZ64I 122648649 IC50 = 6.3 nM T65755 C3Q6FV 127024856 IC50 = 1900 nM T65755 C1WH5M 127024973 IC50 = 139 nM T65755 C8FOZ4 127025172 IC50 > 10000 nM T65755 CE4CI8 127025178 IC50 = 15 nM T65755 CL8TF5 127025475 IC50 > 10000 nM T65755 C8VEY9 127025539 IC50 > 10000 nM T65755 CNSO40 127025540 IC50 = 980 nM T65755 CF4G7Q 127025769 IC50 > 10000 nM T65755 CIF74W 127025777 IC50 > 10000 nM T65755 CT2EK9 127025778 IC50 > 10000 nM T65755 CMWO84 127025780 IC50 > 10000 nM T65755 C43JUF 127026070 IC50 = 1340 nM T65755 C71TBA 127026107 IC50 = 217000 nM T65755 CF4O7N 127026108 IC50 = 786000 nM T65755 CA6Z0B 127026109 IC50 = 84200 nM T65755 CI72YM 127026110 IC50 = 122000 nM T65755 CQ32BA 127026381 IC50 > 10000 nM T65755 CQTF36 127026436 IC50 > 10000 nM T65755 C3Q8FL 127026437 IC50 > 10000 nM T65755 C2N1UD 127026438 IC50 > 10000 nM T65755 CWY63G 127026695 IC50 = 81 nM T65755 CO4JI5 127026735 IC50 = 160 nM T65755 CME4B7 127026736 IC50 = 300 nM T65755 CG34KC 127026737 IC50 = 80 nM T65755 CNX10Q 127026738 IC50 = 1200 nM T65755 CJ0AI5 127026739 IC50 = 170 nM T65755 C60DIS 127026740 IC50 > 10000 nM T65755 C31UJC 127026741 IC50 > 10000 nM T65755 COI3S8 127026742 IC50 = 660 nM T65755 CCR4M7 127026743 IC50 = 400 nM T65755 C4HW8S 127027008 IC50 = 840 nM T65755 C0BG8P 127027017 IC50 = 43 nM T65755 C1EW7J 127027019 IC50 = 1255 nM T65755 C9V1YZ 127027020 IC50 = 715 nM T65755 C1R4SF 127027021 IC50 = 364 nM T65755 CT3Y6R 127027064 IC50 = 132 nM T65755 CI42FJ 127027065 IC50 = 11 nM T65755 CZR43H 127027067 IC50 = 810 nM T65755 CA1N7Y 127027068 IC50 = 2100 nM T65755 CE8CN3 127027069 IC50 = 3100 nM T65755 CCG30L 127027070 IC50 = 540 nM T65755 CU84JL 127027071 IC50 > 10000 nM T65755 CB2F4S 127027091 IC50 = 29 nM T65755 CO3A7W 127027092 IC50 = 8.5 nM T65755 C90VAW 127027093 IC50 = 128 nM T65755 CO9I6S 127027094 IC50 = 29 nM T65755 CFY28V 127027095 IC50 = 18 nM T65755 CGE73Y 127027096 IC50 = 698 nM T65755 CT5VX3 127027322 IC50 > 10000 nM T65755 C6ZX2Y 127027370 IC50 = 3.2 nM T65755 CT2YZ6 127027371 IC50 = 74 nM T65755 CE2LV9 127027372 IC50 = 31 nM T65755 CCXA80 127027373 IC50 = 8.8 nM T65755 CJAE38 127027376 IC50 > 10000 nM T65755 C86OFN 127027393 IC50 > 10000 nM T65755 C8X6FT 127027394 IC50 > 10000 nM T65755 CK0J7H 127027395 IC50 > 10000 nM T65755 CTP3J4 127027396 IC50 > 10000 nM T65755 CJ8MQ3 127027677 IC50 = 23 nM T65755 CK53WF 127027678 IC50 = 150 nM T65755 C3EWH4 127027679 IC50 = 56 nM T65755 C1KWD3 127027680 IC50 = 102 nM T65755 CV2AY4 127027714 IC50 = 545 nM T65755 CM3SZ5 127027716 IC50 = 2200 nM T65755 CM42UC 127027717 IC50 = 1500 nM T65755 CBMZ67 127027718 IC50 = 8600 nM T65755 C1KVR2 127027719 IC50 > 10000 nM T65755 CW8F7D 127027975 IC50 = 3000 nM T65755 C2QYV5 127027979 IC50 = 690 nM T65755 CX80AH 127027993 IC50 = 608 nM T65755 CO5E1V 127027994 IC50 = 102 nM T65755 CG8NU7 127027995 IC50 = 8 nM T65755 CHLF80 127028028 IC50 = 68 nM T65755 CY5OQ9 127028029 IC50 = 12 nM T65755 CZ7C3D 127028030 IC50 = 2.2 nM T65755 CL0W8U 127028035 IC50 = 673 nM T65755 C7PX3L 127028036 IC50 = 554 nM T65755 C39IBG 127028037 IC50 = 145 nM T65755 CD5I1F 127028038 IC50 = 32 nM T65755 CLN54U 127028295 IC50 = 690 nM T65755 CG91JU 127028631 IC50 = 3200 nM T65755 CSI54T 127028894 IC50 = 3700 nM T65755 CV07OM 127028943 IC50 = 18 nM T65755 C08RCM 127028973 IC50 = 33 nM T65755 C8FNI2 127029515 IC50 > 10000 nM T65755 CNP78W 127029538 IC50 = 495000 nM T65755 C40GCD 127029539 IC50 = 188000 nM T65755 CV9I8D 127030313 IC50 = 1500 nM T65755 CR0P1O 127031793 IC50 = 2500 nM T65755 CN53LR 127034811 IC50 = 5960000 nM T65755 CO0W2P 127035816 IC50 = 2330000 nM T65755 CUFI57 127035817 IC50 = 2190000 nM T65755 CL98ZS 127035818 IC50 = 4370000 nM T65755 CH8JV6 127035819 IC50 = 4260000 nM T65755 CYF2I3 127035820 IC50 = 1660000 nM T65755 C9AJ6H 127035854 IC50 = 3740000 nM T65755 CGP2L9 127035988 IC50 = 2680000 nM T65755 CHPK02 127035989 IC50 = 290000 nM T65755 CIE4D3 127035990 IC50 = 970000 nM T65755 C8ZRA0 127035991 IC50 = 450000 nM T65755 CHQ46B 127035993 IC50 = 3460000 nM T65755 C9FKB5 127037004 IC50 = 3200000 nM T65755 CBG31X 127037135 IC50 = 2940000 nM T65755 CPH6Q8 127038650 IC50 = 810 nM T65755 CU1JM3 127038651 IC50 = 1170 nM T65755 CUR0C1 127038652 IC50 = 2240 nM T65755 C18FSM 127039340 IC50 = 270 nM T65755 CIO0G3 127039341 IC50 = 350 nM T65755 C0D1HL 127039342 IC50 = 820 nM T65755 C4Q7YV 127039343 IC50 = 3160 nM T65755 C12NJF 127039347 IC50 = 510 nM T65755 CGK1P6 127039348 IC50 = 860 nM T65755 CFU02P 127039661 IC50 = 1330 nM T65755 C8C0SL 127039665 IC50 = 1050 nM T65755 C9WLF2 127039908 IC50 = 1430 nM T65755 C69IXG 127041845 IC50 = 430 nM T65755 CLQH35 127042561 IC50 = 6170 nM T65755 CP9AI0 127042572 IC50 = 1430 nM T65755 CPX13Q 127042871 IC50 = 1810 nM T65755 CJ72GX 127042872 IC50 = 2450 nM T65755 CZV43J 134283792 IC50 = 53000 nM T65755 CO7K3N 134283799 IC50 = 14000 nM T65755 C1Y4TA 134283810 IC50 = 60000 nM T65755 CV2YF7 134283813 IC50 = 62000 nM T65755 CI28ZH 135424818 EC50 = 148 nM T65755 C01EZF 135567459 IC50 = 54000 nM T65755 CFHE27 135906525 EC50 = 2090 nM T65755 CHY18X 135906526 EC50 = 7890 nM T65755 CU3BA9 135906527 EC50 = 125000 nM T65755 CDOM93 135906528 EC50 = 4160 nM T65755 C8M6LX 135906529 EC50 = 6630 nM T65755 CU64IM 135906530 EC50 = 2080 nM T65755 C93OEC 135906531 EC50 = 177 nM T65755 C70LDS 135906532 EC50 = 474 nM T65755 CG63ID 135985827 IC50 = 105 nM T65755 CP56QS 135985828 IC50 = 178 nM T65755 C1OS6C 135985829 IC50 = 41 nM T65755 CZ92NX 135985856 IC50 = 23 nM T65755 CB3U5Z 135985857 IC50 = 86 nM T65755 CLBO25 135985864 IC50 = 333 nM T65755 CUP57J 135985865 IC50 = 49 nM T65755 CMTH01 135985866 IC50 = 219 nM T65755 CD9U8W 136002521 IC50 > 100000 nM T65755 C50ZPJ 136007828 IC50 = 22 nM T65755 CZQ4E3 136007829 IC50 = 18 nM T65755 C4S3PX 136007831 IC50 = 62 nM T65755 C95PVG 136007832 IC50 = 77 nM T65755 CIVE47 136015315 IC50 = 55 nM T65755 CT7Q8M 136015316 IC50 = 132 nM T65755 CEP24G 136015317 IC50 = 137 nM T65755 CTCM97 136015318 IC50 = 838 nM T65755 C17BPS 136015319 IC50 = 54 nM T65755 C8VB1S 136015320 IC50 = 115 nM T65755 C3ANQ8 136015321 IC50 = 90 nM T65755 C0BM3W 136015322 IC50 = 171 nM T65755 CC68RY 136015323 IC50 = 403 nM T65755 CXJ03M 136015324 IC50 = 510 nM T65755 C2WR6A 136015325 IC50 = 111 nM T65755 C0X9OV 136015326 IC50 = 94 nM T65755 C0OLS8 136030779 IC50 = 37000 nM T65755 CIA7R4 136030780 IC50 = 23000 nM T65755 C24LKN 136030781 IC50 = 44000 nM T65755 C85OIV 136069550 IC50 = 4 nM T65755 CM58ET 136069551 IC50 = 19 nM T65755 CD12MQ 136069552 IC50 = 140 nM T65755 CPNB26 136069553 IC50 = 7 nM T65755 C5HY9J 136069558 IC50 = 31 nM T65755 C82ZAV 136069559 IC50 = 5 nM T65755 C35ZKT 136136549 IC50 > 100000 nM T65755 CTFI74 136184410 EC50 = 186 nM T65755 CSP1N0 136184411 EC50 = 250 nM T65755 C0TZP5 136184412 EC50 = 291 nM T65755 CU3AH7 136184413 EC50 = 763 nM T65755 C46KWH 136184414 EC50 = 3790 nM T65755 CDR9X0 137174935 IC50 = 70 nM T65755 C75MCW 137487425 IC50 = 11300 nM T65755 C5LM0P 137487426 IC50 > 20000 nM T65755 C0MV4B 137487427 IC50 = 3000 nM T65755 C3LUJ0 137487429 IC50 = 1400 nM T65755 CT2H1X 137487451 IC50 > 20000 nM T65755 CK92LE 137487458 IC50 > 20000 nM T65755 C9ONI5 137629006 IC50 = 3000 nM T65755 CVG3D0 137629277 IC50 = 270 nM T65755 C2YL4I 137629294 IC50 = 21000 nM T65755 CL6ON4 137629786 IC50 = 9000 nM T65755 CXV84M 138377596 IC50 = 2 nM T65755 CIWG23 138393067 IC50 = 4600 nM T65755 CC0B6V 140846804 IC50 = 3300 nM T65755 CP73QO 141504704 IC50 = 8700 nM T65755 CFZ80E 141504707 IC50 > 20000 nM T65755 CTON95 141504712 IC50 = 19000 nM T65755 CV9C7B 141504714 IC50 = 5000 nM T65755 C4WK5N 141504719 IC50 = 15100 nM T65755 CX7KL4 141504721 IC50 > 20000 nM T65755 C9D3OI 141504722 IC50 = 3000 nM T65755 CQ04HU 141504728 IC50 = 21300 nM T65755 CEHD51 141728806 IC50 = 19 nM T65755 CCY30N 141728810 IC50 > 10000 nM T65755 CLH76T 141728811 IC50 = 37 nM T65755 CQB0U4 141728813 IC50 = 3 nM T65755 CN75MA 141728817 IC50 = 2 nM T65755 CWN43D 141728825 IC50 = 41 nM T65755 C7FW8A 141728827 IC50 = 4 nM T65755 CHS9N0 141728829 IC50 = 62 nM T65755 CN72IC 141728831 IC50 = 3 nM T65755 C7EL5X 141728840 IC50 = 13 nM T65755 C9H8PX 141728841 IC50 = 20 nM T65755 CBV2K5 141728842 IC50 = 15 nM T65755 CZ8J7C 141728843 IC50 > 10000 nM T65755 C2HF9A 141728845 IC50 = 38 nM T65755 CBRN42 141728846 IC50 = 10 nM T65755 COEV20 141728855 IC50 = 3 nM T65755 CC03XH 141728860 IC50 = 40 nM T65755 C4RGY1 141728867 IC50 = 569 nM T65755 CNUG79 141728871 IC50 = 26 nM T65755 C65GLX 141728873 IC50 = 26 nM T65755 C9IW0F 141728874 IC50 = 37 nM T65755 C18SJO 141728877 IC50 = 18 nM T65755 CJRV01 145949203 IC50 = 370 nM T65755 CS72AE 145951731 IC50 = 520 nM T65755 CHA86R 145952233 IC50 = 550 nM T65755 CM53ZB 145954785 IC50 = 560 nM T65755 CXR4K9 145956541 IC50 = 292000 nM T65755 CJ86KW 145957429 IC50 = 410 nM T65755 CZ6L7T 145964935 IC50 = 820 nM T65755 CTUF34 145966712 IC50 = 3.3 nM T65755 CJFP12 145966738 IC50 = 25 nM T65755 C93JKN 145967593 IC50 = 1439 nM T65755 CD82XB 145967610 IC50 = 16 nM T65755 C7OG1D 145967698 IC50 = 1460 nM T65755 CEXK31 145967726 IC50 = 22.2 nM T65755 C5RPQ9 145967832 IC50 = 33 nM T65755 CI1ZD2 145967851 IC50 = 3827 nM T65755 CR59HK 145967905 IC50 = 644 nM T65755 C95SNQ 145967968 IC50 = 1139 nM T65755 CX0OD9 145968046 IC50 = 8.1 nM T65755 CES7W6 145968087 IC50 = 1792 nM T65755 C79TFD 145968094 IC50 = 59.5 nM T65755 CW87FU 145968130 IC50 = 268.9 nM T65755 CR2D4Y 145968170 IC50 = 7.6 nM T65755 C4M7TF 145968305 IC50 = 22.5 nM T65755 CSO4I7 145968364 IC50 > 5000 nM T65755 C2XS8E 145968675 IC50 = 74 nM T65755 CI0JR2 145968743 IC50 = 29.5 nM T65755 CG0S9U 145968824 IC50 = 1028 nM T65755 C49PHB 145968907 IC50 = 112.1 nM T65755 CIA79M 145968985 IC50 = 40 nM T65755 CQUJ51 145969013 IC50 = 311.9 nM T65755 C9DNC2 145969078 IC50 = 165.5 nM T65755 C2M4KV 145969297 IC50 = 36.9 nM T65755 CS8AI5 145969319 IC50 = 249.1 nM T65755 C27YHM 145969456 IC50 = 43 nM T65755 CV53YN 145969651 IC50 = 165 nM T65755 C2XOW7 145969735 IC50 = 21.8 nM T65755 C0K6XS 145969789 IC50 = 22 nM T65755 CUI37A 145969799 IC50 = 2 nM T65755 CZ80EP 145969996 IC50 = 231 nM T65755 C1VM0B 145970100 IC50 = 57.1 nM T65755 C94FBQ 145970117 IC50 = 84.8 nM T65755 C7TSV2 145970161 IC50 = 2603 nM T65755 CG5OK8 145970171 IC50 = 58 nM T65755 CBR60K 145970453 IC50 = 476 nM T65755 C3D9LJ 145970457 IC50 = 2 nM T65755 C0E2UO 145970598 IC50 = 22 nM T65755 C0Z7IU 145970680 IC50 = 35.8 nM T65755 CRW0X3 145970971 IC50 > 20000 nM T65755 CPF8G7 145971126 IC50 = 37.3 nM T65755 C61IRF 145974167 IC50 = 680 nM T65755 C3BM7K 145974717 IC50 = 17 nM T65755 CN4E5O 145976956 IC50 = 180 nM T65755 CZ19QM 145977548 IC50 = 19800 nM T65755 C7X4LZ 145978932 IC50 = 1800 nM T65755 CSA0K9 145979160 IC50 = 370 nM T65755 CDG5U8 145980347 IC50 = 930 nM T65755 CS80AL 145980924 IC50 = 2820 nM T65755 CW6US1 145981665 IC50 = 260 nM T65755 C9VDE5 145982499 IC50 = 86.9 nM T65755 C6OL1K 145983267 IC50 = 862.9 nM T65755 C8O1GU 145983616 IC50 > 10000 nM T65755 C17UTC 145983813 IC50 > 10000 nM T65755 CIWO70 145984314 IC50 = 174.4 nM T65755 C9ZKC1 145984665 IC50 = 104.7 nM T65755 CN6KB9 145985243 IC50 = 61.2 nM T65755 CB24HO 145985400 IC50 = 720 nM T65755 C1WH7V 145986586 IC50 > 5000 nM T65755 C7L1GU 145986811 IC50 = 5.7 nM T65755 CRX8H1 145987492 IC50 = 13 nM T65755 CPAX89 145987732 IC50 = 8 nM T65755 CV8LF0 145987823 IC50 = 850 nM T65755 CH7I5Z 145988992 IC50 = 5630 nM T65755 CTK67P 145989067 IC50 = 230 nM T65755 CJ8DO3 145989487 IC50 = 121 nM T65755 CO4J2D 145990209 EC50 = 350 nM T65755 C1E8IF 145990399 IC50 = 4780 nM T65755 C58OZE 145990872 IC50 = 830 nM T65755 CB0C7M 145991220 IC50 = 1750 nM T65755 CR2Q5I 145991323 IC50 = 27750 nM T65755 CQ4TP0 145992467 IC50 = 340 nM T65755 C5UP4V 145993239 IC50 > 100000 nM T65755 CQ4GW3 145993428 IC50 = 960 nM T65755 C3M4ND 145993768 IC50 = 2690 nM T65755 C2ST6R 145993977 IC50 = 5735 nM T65755 C1W6CF 145994016 IC50 = 65000 nM T65755 C8ZB6S 145994163 IC50 = 3060 nM T65755 C3SA6B 148608442 IC50 = 71.5 nM T65755 CO47EC 148970856 IC50 = 132.6 nM T65755 CZ0LP6 150496562 IC50 = 18 nM T65755 CO5BV8 155510418 IC50 = 80 nM T65755 CV1UX5 155510762 IC50 = 900 nM T65755 CJ2KD4 155512410 IC50 = 40 nM T65755 C0ZN3E 155512623 IC50 = 11600 nM T65755 C7VKU2 155513116 IC50 = 10720 nM T65755 CA2LG5 155513254 IC50 = 1920 nM T65755 CLAY24 155513547 IC50 = 7650 nM T65755 CE9RZ2 155513746 IC50 = 2770 nM T65755 C6BV9W 155514532 IC50 = 4330 nM T65755 C2UJ1K 155515909 IC50 = 144000 nM T65755 CT8XU7 155516547 IC50 = 210 nM T65755 CP57FO 155517042 IC50 = 2290 nM T65755 C7G0XM 155517418 IC50 = 3150 nM T65755 CCDU61 155518496 IC50 > 32000 nM T65755 C94VUT 155518725 IC50 = 6850 nM T65755 CDY5H6 155519645 IC50 = 360820 nM T65755 CG4F2U 155521283 IC50 > 32000 nM T65755 CAR0O8 155521402 IC50 = 8310 nM T65755 C82PHV 155521822 IC50 = 6820 nM T65755 C4FS3Y 155521883 IC50 = 130 nM T65755 C6DVZ9 155521965 IC50 = 4480 nM T65755 CJ3E4G 155524660 IC50 = 22800 nM T65755 CQ3AI0 155525851 IC50 = 211330 nM T65755 CH52FD 155526273 IC50 = 105470 nM T65755 CW2H5R 155527295 IC50 = 180 nM T65755 C71UNO 155527385 IC50 = 270 nM T65755 CQK19H 155527955 IC50 = 1010 nM T65755 C6R9TE 155528027 IC50 = 280 nM T65755 CLVW69 155528303 IC50 > 1000000 nM T65755 C5F1IZ 155528743 IC50 > 1000000 nM T65755 C9TIO5 155528896 IC50 = 391400 nM T65755 C2SXP9 155529646 IC50 = 940 nM T65755 C94BFW 155529690 IC50 = 21900 nM T65755 CO8Q9P 155530125 IC50 = 1810 nM T65755 C1B2FN 155530610 IC50 = 126010 nM T65755 C76BIC 155531415 IC50 = 3150 nM T65755 CUC3P1 155531533 IC50 = 3930 nM T65755 CL0W5T 155531877 IC50 = 1 nM T65755 C0VZ9J 155532068 IC50 = 415070 nM T65755 CH27XY 155536857 IC50 = 3530 nM T65755 C81KIF 155537008 IC50 = 990 nM T65755 C2JH0S 155537112 IC50 = 110 nM T65755 CTF70E 155537700 IC50 = 270 nM T65755 CS12HW 155538841 IC50 = 46 nM T65755 CLD19W 155539311 IC50 = 194550 nM T65755 CT04NP 155540027 IC50 = 970 nM T65755 CUZV73 155540466 EC50 = 8140 nM T65755 CQX12L 155541458 IC50 = 150 nM T65755 C7B5NU 155541992 IC50 = 13000 nM T65755 CAM3C1 155542624 IC50 = 3000 nM T65755 COF0D1 155542875 IC50 = 1570 nM T65755 C01SCV 155543375 IC50 = 1980 nM T65755 CKJ03M 155543455 IC50 = 4030 nM T65755 C5ENC1 155543511 IC50 = 3340 nM T65755 CP6Q8B 155544130 IC50 = 4500 nM T65755 CM6HT8 155544609 IC50 = 1120 nM T65755 CS1P3J 155545401 IC50 = 671830 nM T65755 CH6J1X 155545613 IC50 = 150 nM T65755 CPE37N 155546987 IC50 = 92 nM T65755 C1D4PI 155547606 IC50 = 490 nM T65755 CF64DP 155547817 IC50 = 4650 nM T65755 CRLE97 155547991 IC50 = 90 nM T65755 CQ2FB6 155548396 IC50 = 170 nM T65755 C9WJ4G 155548562 IC50 = 260 nM T65755 C7CXL4 155548945 IC50 = 260 nM T65755 CTFU61 155549051 IC50 = 830 nM T65755 CD8B2Q 155549392 IC50 = 1120 nM T65755 C02YXA 155550058 IC50 = 461700 nM T65755 CO6ID4 155550122 IC50 = 144 nM T65755 C16FOI 155550728 IC50 = 170 nM T65755 CU3Y5K 155551054 IC50 = 10 nM T65755 C4Q7CM 155551213 IC50 = 470 nM T65755 CEO4J8 155551917 IC50 = 19 nM T65755 C6FW7Z 155552055 IC50 = 120 nM T65755 CTM6B4 155553047 IC50 = 240 nM T65755 CWBP87 155553299 IC50 = 120 nM T65755 C7PBK3 155553376 IC50 = 6800 nM T65755 C49VRW 155554090 IC50 = 210 nM T65755 C1LE0Z 155554153 IC50 = 230 nM T65755 CL7G8P 155554796 IC50 = 680 nM T65755 CWV2Y0 155556131 IC50 = 850 nM T65755 CG9NP0 155556271 IC50 = 8590 nM T65755 C9Q6MF 155558959 IC50 = 132 nM T65755 C6N2VW 155559068 IC50 = 2700 nM T65755 C2IS1E 155559200 IC50 = 52 nM T65755 C1LK7O 155559569 IC50 = 130 nM T65755 CPD50Q 155559583 EC50 = 7840 nM T65755 CC62UI 155559872 IC50 = 470 nM T65755 CR9F7Q 155560385 IC50 = 3140 nM T65755 C1T8VS 155560660 IC50 = 40300 nM T65755 C41QXD 155560908 IC50 = 1860 nM T65755 C01FJW 155561174 IC50 = 150 nM T65755 CYL48D 155561445 IC50 = 3140 nM T65755 C8HN2B 155563943 IC50 = 104 nM T65755 C9UYZ6 155564157 IC50 = 35 nM T65755 C49QWP 155564188 IC50 = 73 nM T65755 CR85ZW 155564587 IC50 = 4130 nM T65755 C9F6VR 155564907 IC50 = 200 nM T65755 CH9CU3 155566324 IC50 = 400 nM T65755 C51BFK 155566644 IC50 = 630 nM T65755 CT6Z4H 155567814 IC50 = 62 nM T65755 CUA7B3 155568680 IC50 = 300 nM T65755 CLFT12 155568761 IC50 = 30 nM T65755 CF2X0U 155568767 IC50 = 4940 nM T65755 CQ4GX2 155569054 IC50 = 560 nM T65755 C5NQK8 155569352 IC50 = 77 nM T65755 CZVT07 44422818 IC50 = 8100 nM T65755 D00DQZ 11964504 IC50 = 81 nM T65755 D00HFS 46884057 IC50 = 30 nM T65755 D00KFF 9882812 IC50 = 6700 nM T65755 D00PLM 44418106 IC50 = 1130 nM T65755 D00SEE 11379392 IC50 = 58 nM T65755 D00ZSD 11694528 IC50 = 7700 nM T65755 D01EDB 135903324 IC50 = 104 nM T65755 D01FYB 23648267 IC50 = 3000 nM T65755 D01LDQ 24749070 IC50 = 5000 nM T65755 D01MFV 44401339 IC50 = 12500 nM T65755 D01XWZ 11220728 IC50 = 1100 nM T65755 D01XXN 11196500 IC50 = 110 nM T65755 D02HCQ 1794427 Ki = 135 nM T65755 D02HVH 11427204 IC50 = 170 nM T65755 D02MQM 9927379 IC50 = 17000 nM T65755 D02UTC 11323577 IC50 = 2500 nM T65755 D02WZK 44350626 IC50 = 1100 nM T65755 D03QOD 239512 IC50 = 4600 nM T65755 D03XXI 44341224 IC50 = 3700 nM T65755 D04DOL 25032059 IC50 = 50 nM T65755 D04GGW 10967421 IC50 = 306 nM T65755 D04HSS 11447748 IC50 = 360 nM T65755 D04LLD 22915465 IC50 = 20 nM T65755 D04NSP 11086699 IC50 = 149 nM T65755 D04ZDI 11231829 IC50 = 68 nM T65755 D05AHZ 11572583 IC50 = 40 nM T65755 D05GVY 11254470 IC50 = 7100 nM T65755 D05LLX 11287488 IC50 = 1500 nM T65755 D05PYF 10242569 IC50 = 243 nM T65755 D05VFP 44350703 IC50 = 520 nM T65755 D05XAN 11449823 IC50 = 75 nM T65755 D06IMY 44626296 IC50 = 3000 nM T65755 D06IQB 3082127 IC50 = 450 nM T65755 D06VBN 11347053 IC50 = 54 nM T65755 D06XNP 11277483 IC50 = 610 nM T65755 D07FJU 11345433 IC50 = 110 nM T65755 D08PMD 9921260 IC50 = 238 nM T65755 D09LVY 11964503 IC50 = 150 nM T65755 D09SUO 5269 IC50 > 75000 nM T65755 D09YBN 11298778 IC50 = 11000 nM T65755 D09ZNU 11817702 IC50 = 210 nM T65755 D0A5LS 403373 IC50 = 369 nM T65755 D0A7IF 44418125 IC50 = 1260 nM T65755 D0AX7B 44341053 IC50 = 2900 nM T65755 D0B2ZJ 44350718 IC50 = 620 nM T65755 D0B3ZM 11436024 IC50 = 370 nM T65755 D0C0VP 23327627 IC50 = 17000 nM T65755 D0C2KD 9943996 IC50 = 1556 nM T65755 D0D2KE 11608171 IC50 = 6200 nM T65755 D0D3XC 11708207 IC50 = 2170 nM T65755 D0E1QP 4262314 IC50 > 100000 nM T65755 D0E8KR 11747496 IC50 = 248 nM T65755 D0F0KS 44401305 IC50 = 2800 nM T65755 D0FN5D 45482672 IC50 = 3500 nM T65755 D0H1FZ 24759251 IC50 = 9600 nM T65755 D0H7QA 46884056 IC50 = 30 nM T65755 D0I4RK 45482660 IC50 = 16000 nM T65755 D0KE3I 44350655 IC50 = 990 nM T65755 D0L6YF 46884016 IC50 = 32 nM T65755 D0M0QJ 10452725 IC50 = 29 nM T65755 D0P1HZ 6917986 IC50 = 2 nM T65755 D0Q2CC 46884055 IC50 = 251 nM T65755 D0Q5MC 24753719 IC50 > 100000 nM T65755 D0Q8QA 44418141 IC50 = 750 nM T65755 D0QO0L 11312563 IC50 = 34 nM T65755 D0R2HF 11437457 IC50 = 390 nM T65755 D0R5VG 11472431 IC50 = 250 nM T65755 D0RU1X 298878 IC50 = 270 nM T65755 D0S7WQ 9994848 IC50 = 44 nM T65755 D0S9JF 11637291 IC50 = 120 nM T65755 D0T2QL 444539 Ki = 8.21 nM T65755 D0T4IY 10379373 IC50 = 72 nM T65755 D0T4JQ 264 Ki = 136000 nM T65755 D0V2ZO 11528707 IC50 = 2580 nM T65755 D0V9EN 689043 Ki = 10840 nM T65755 D0W1PV 6918328 IC50 = 0.004 ug.mL-1 T65755 D0X1CB 395803 IC50 < 5 nM T65755 D0X4VO 44359538 IC50 > 100000 nM T65755 D0XZ9Q 11149404 IC50 = 1500 nM T65755 D0YO6M 785232 IC50 = 3000 nM T65755 D0YP4F 10383069 IC50 = 6.6 nM T65755 D0YY9M 9965141 IC50 = 1006 nM T65755 D0Z2GH 44563351 IC50 = 22 nM T65755 D0Z3BM 44342825 IC50 = 2600 nM T65755 D0Z5KX 11346934 IC50 = 340 nM T65755 D0Z7YS 44361923 IC50 = 3600 nM T84439 CJB93K 1555702 EC50 = 162 nM T84439 CW2Z0P 2109722 EC50 = 32 nM T84439 CTM14Y 2303171 EC50 = 150 nM T84439 C40EUH 2548543 EC50 = 2100 nM T84439 CO78IS 2548547 EC50 = 16 nM T84439 CHP01V 2856847 EC50 = 670 nM T84439 CM6G3H 3376937 EC50 = 43 nM T84439 C41YLH 7534868 EC50 = 24 nM T84439 CZ5K4W 26532940 EC50 = 118 nM T84439 C9PM7R 28821961 EC50 = 54 nM T84439 CPE3W0 28918445 EC50 = 33 nM T84439 CNAU92 28918448 EC50 = 1700 nM T84439 C4XEG5 40719079 EC50 = 193 nM T84439 CAW21Y 122195499 EC50 = 66 nM T84439 CPB8M1 122195500 EC50 = 440 nM T84439 C68YAH 122195501 EC50 = 283 nM T84439 CL4G6O 122195502 EC50 = 10000 nM T84439 C7UD6N 122195638 EC50 = 59 nM T84439 CP96TA 122195639 EC50 = 52 nM T84439 CWC1F8 122195640 EC50 = 46 nM T84439 CY7TE4 122195641 EC50 = 52 nM T84439 CCJS89 122195642 EC50 = 40 nM T84439 CR2F1S 122195643 EC50 = 46 nM T84439 CJ7L8U 122195644 EC50 = 24 nM T84439 C8BCA0 122195645 EC50 = 78 nM T84439 C4K9RJ 122195646 EC50 > 10000 nM T84439 CNV39B 122195647 EC50 > 10000 nM T53510 CG4P6H 4411483 IC50 = 19100 nM T53510 C7EOJ1 9812342 IC50 = 5 nM T53510 C06ENG 44385619 IC50 = 90000 nM T53510 CAZ2K0 44385682 IC50 = 220000 nM T53510 C7HWG6 44385932 IC50 = 4100 nM T53510 CQ7V5J 44386040 IC50 = 66000 nM T53510 C6IM9P 44386041 IC50 = 41000 nM T53510 CAGC58 44386723 IC50 = 8400 nM T53510 C0W2HB 44386941 IC50 = 48000 nM T53510 CIS37G 44386993 IC50 = 143300 nM T53510 CS9HI5 44387048 IC50 > 250000 nM T53510 C3G1TO 44387218 IC50 = 31900 nM T53510 CY0KD5 44597665 IC50 > 100000 nM T53510 CP1YM8 56926704 IC50 > 100000 nM T53510 CKR36B 56926707 IC50 > 100000 nM T53510 C0IV7W 56926708 IC50 > 100000 nM T53510 CYC1M7 56926806 IC50 > 100000 nM T53510 CQH63T 56926807 IC50 = 77600 nM T53510 C2VQ0R 56926808 IC50 = 96300 nM T53510 C98YWR 56926809 IC50 = 93000 nM T53510 C40ALR 56926915 IC50 = 178600 nM T53510 C40KLT 56926916 IC50 = 94200 nM T53510 CQXL53 56926917 IC50 = 66300 nM T53510 C0C9PN 56926918 IC50 = 33100 nM T22118 D01AZG 5073 Ki = 21 nM T22118 D01FFA 72301 Ki = 153 nM T22118 D01ZII 2726 Ki = 96 nM T22118 D03KQF 4011 Ki = 402 nM T22118 D04JCN 47811 Ki = 2020 nM T22118 D04JEE 4946 EC50 > 5011.87 nM T22118 D05XGO 11154555 Ki = 2100 nM T22118 D0B0CP 667467 Ki = 18 nM T22118 D0CQ0Z 33630 Ki = 147 nM T22118 D0D1AL 3559 Ki = 6.166 nM T22118 D0G8NN 119570 Ki > 10000 nM T22118 D0H3HM 60795 Ki = 310 nM T22118 D0H6QU 6005 EC50 = 3.77 nM T22118 D0H7KF 5002 Ki = 390 nM T22118 D0I8FI 3779 Ki > 50000 nM T22118 D0KS6W 7077 Ki = 343 nM T22118 D0P5SA 3372 Ki = 179 nM T22118 D0R1JV 60854 Ki = 9.5 nM T22118 D0R6BI 3341 EC50 = 2.8 nM T22118 D0R9EQ 5095 Ki = 32500 nM T22118 D0T6QX 5736 Ki = 29 nM T22118 D0T7OW 681 EC50 = 20 nM T22118 D0V4QS 135398745 Ki = 10 nM T22118 D0X7KB 28864 Ki = 77 nM T22118 D0Y5UG 2160 Ki = 89 nM T22118 D0Z1RV 135398737 Ki = 7.5 nM T22118 D0K7ZH 86764100 Ki = 8.54 nM T22118 D0LI1C 44469321 IC50 > 10000 nM T22118 D0N1HW 5311200 Ki > 10000 nM T22118 D0Y6HW 107930 Ki = 1.2 nM T22118 D07YLK 4350931 Ki = 1.862 nM T22118 D0NH9P 135 EC50 = 1.11 nM T22118 D01RAE 133079 Ki > 8378 nM T22118 D01WJZ 60820 Ki > 5000 nM T22118 D02DHU 1218 EC50 = 4.7 nM T22118 D06DZI 107780 Ki < 10000 nM T22118 D09DRG 9952420 IC50 > 10000 nM T22118 D0EE6L 3038495 Ki = 760 nM T22118 D0N1WM 122324 EC50 = 1.95 nM T22118 D0OS6O 60149 Ki = 210 nM T22118 D0OU7P 1242 EC50 = 1.1 nM T22118 D0OW1R 9802631 Ki > 10000 nM T22118 D0P2YS 6603703 EC50 = 3 nM T22118 D0ZG9N 132337 Ki > 10000 nM T22118 C7DT6H 15115517 Ki = 130 nM T22118 CY9E4K 15115518 Ki = 170 nM T22118 C41ZLR 1225 EC50 = 0.73 nM T22118 C7ALK2 1240 Ki = 804 nM T22118 CUB9O5 1241 EC50 = 1 nM T22118 CZUI83 2769 IC50 = 1700 nM T22118 CW56ZA 5290 Ki = 5.6 nM T22118 C5H9CN 9287 Ki > 10000 nM T22118 CVW5J9 10220 Ki = 15 nM T22118 CRD7M3 11492 Ki = 48000 nM T22118 C9E6DA 21171 Ki = 48.6 nM T22118 C17TDE 23269 Ki > 10000 nM T22118 COI7E6 59227 EC50 = 28 nM T22118 C1PT7R 64638 EC50 = 5.1 nM T22118 CBJ5R0 65340 EC50 = 37 nM T22118 C6CU1T 70515 Ki > 10000 nM T22118 CPZ5N6 98358 Ki > 10000 nM T22118 C9NJK8 114876 Ki > 10000 nM T22118 C9VZR2 121852 IC50 = 39810.72 nM T22118 CN9X8Q 122132 Ki = 5400 nM T22118 CG21YH 127262 Ki = 207 nM T22118 CV48UJ 130424 Ki = 6 nM T22118 CZIL53 130844 Ki = 0.9 nM T22118 CY8W6U 131213 Ki > 5000 nM T22118 CS8W1F 133642 EC50 = 717.5 nM T22118 CZL87W 133999 IC50 > 10000 nM T22118 COJK09 146266 EC50 = 40.4 nM T22118 C7I3TL 147514 Ki = 1.1 nM T22118 C1ND9W 161665 Ki = 50 nM T22118 C9OD2N 163091 Ki = 8.9 nM T22118 CLK7P3 169713 IC50 > 10000 nM T22118 CXS17Y 188442 Ki = 530 nM T22118 C2INS1 201536 EC50 = 20.4 nM T22118 C5RC4G 231915 Ki > 10000 nM T22118 CYO3R2 300430 Ki > 10000 nM T22118 CAH2S5 439654 Ki = 22 nM T22118 CG2JX9 440229 Ki = 4.5 nM T22118 C56WSX 443422 Ki > 5000 nM T22118 CHB7D2 453215 IC50 = 410 nM T22118 CD7P8Y 763194 Ki > 10000 nM T22118 C6QLR0 763343 Ki > 10000 nM T22118 CLR75J 763625 Ki > 10000 nM T22118 C5SXQ1 763774 Ki > 10000 nM T22118 C9IK2J 792265 Ki > 10000 nM T22118 C13TYL 792460 Ki > 10000 nM T22118 C4AY9X 792584 Ki > 10000 nM T22118 CJ3H2X 1152279 Ki = 529 nM T22118 CVTP62 1811569 Ki > 10000 nM T22118 CT80MF 3033200 EC50 = 31.62 nM T22118 C4TB0I 3036864 Ki = 0.11 nM T22118 C64CZV 3038494 Ki = 1132 nM T22118 CE4KC8 3038603 Ki = 0.3 nM T22118 C54FEG 3039881 Ki = 0.33 nM T22118 CT51WS 3045992 EC50 = 7.943 nM T22118 C82GMT 3246443 Ki = 6.3 nM T22118 C0U6EW 3504099 Ki > 10000 nM T22118 C6AQP8 5249952 Ki = 742 nM T22118 C9AZ2I 5249956 Ki = 3.467 nM T22118 CI45UV 5311428 Ki = 6 nM T22118 C4N7ZW 6101909 Ki = 898 nM T22118 CO3N1A 6440792 Ki = 0.1 nM T22118 CHO8D2 6453963 EC50 = 5.6 nM T22118 CVBX47 6603800 Ki = 192 nM T22118 CIZ7U3 6603820 Ki = 6.2 nM T22118 C6I3MZ 6603954 Ki = 230 nM T22118 CI1CA5 6604773 EC50 = 3.9 nM T22118 C3A1FO 6604789 Ki < 100000 nM T22118 CUN63S 6852375 EC50 = 56 nM T22118 C8QM7B 6852376 Ki = 5.1 nM T22118 C1MHE9 9549058 IC50 = 670 nM T22118 CO5VP3 9796958 EC50 = 1700 nM T22118 C0TX4L 9800145 Ki > 1000 nM T22118 C8XGV3 9804849 IC50 = 900 nM T22118 C9MH4N 9818423 Ki = 8.7 nM T22118 C8NIP0 9819042 Ki = 12 nM T22118 CO9VA3 9820671 IC50 > 1000 nM T22118 CBN06W 9839050 Ki = 63 nM T22118 CS2M1N 9841398 EC50 = 9 nM T22118 C2RQ5H 9843062 Ki > 1000 nM T22118 C7EZ2L 9859861 Ki > 10000 nM T22118 C5WYN4 9865858 Ki > 1000 nM T22118 CQ4LC2 9872676 Ki = 1620 nM T22118 C3DB5H 9884781 Ki > 3000 nM T22118 C9GB2M 9888555 Ki = 670 nM T22118 C6WY0D 9891901 Ki > 10000 nM T22118 CYWQ50 9906447 Ki > 10000 nM T22118 C6CZ3G 9906777 IC50 > 10000 nM T22118 C7SMT0 9908904 IC50 > 1000 nM T22118 C5AHG4 9909521 Ki = 5.5 nM T22118 CO7BK6 9909648 Ki = 411 nM T22118 C4L2CV 9911120 IC50 < 10000 nM T22118 CC6M7Z 9980998 Ki = 2100 nM T22118 CP41ZO 9992499 Ki = 61 nM T22118 CQL12P 10004545 Ki > 2000 nM T22118 C5MUC9 10015045 Ki = 61 nM T22118 C61KDJ 10015860 EC50 = 6.7 nM T22118 C91DQP 10020353 EC50 = 0.12 nM T22118 C2C1XS 10042602 Ki = 4677.35 nM T22118 C4GHO2 10053476 Ki = 1400 nM T22118 C3TJ0U 10066604 Ki > 1000 nM T22118 CI28QJ 10088113 Ki = 0.58 nM T22118 CQVJ58 10088453 Ki = 812.83 nM T22118 CR3D5E 10091430 IC50 = 3311.31 nM T22118 CJXQ40 10092819 Ki = 1100 nM T22118 C5PJ3N 10107367 Ki = 6.607 nM T22118 CZKG96 10200496 Ki = 162 nM T22118 CYT27X 10247457 Ki > 1000 nM T22118 CG2B7I 10247701 Ki = 3981.07 nM T22118 CE9Y8J 10276451 Ki = 1195 nM T22118 CA3E4W 10316297 Ki = 5754.4 nM T22118 CRQN68 10333842 Ki = 45 nM T22118 C3E5CB 10337773 Ki < 100000 nM T22118 CD63EZ 10379766 Ki = 29 nM T22118 C6J2ZL 10402378 Ki = 35.5 nM T22118 C8S3XE 10409556 IC50 = 831.76 nM T22118 C4UN0A 10436653 Ki = 380 nM T22118 C8KD1B 10438027 Ki = 2920 nM T22118 C4LJW3 10452020 Ki = 3 nM T22118 CPI5M7 10476504 Ki = 1500 nM T22118 CEF2O6 10478367 Ki > 10000 nM T22118 C48BRW 10546334 Ki = 3630.78 nM T22118 C9A8KN 10862425 Ki = 2000 nM T22118 CMV36C 10884046 Ki = 1500 nM T22118 CRI50E 10885636 IC50 = 1120 nM T22118 CNP08C 10891703 Ki > 10000 nM T22118 CU80EA 10895106 Ki = 1400 nM T22118 CX65PW 10907460 IC50 = 967 nM T22118 CJC9K4 11005810 IC50 = 376 nM T22118 CB7N1P 11035765 IC50 = 2500 nM T22118 C01NDT 11036640 Ki = 1200 nM T22118 CU6HR7 11036641 Ki = 2200 nM T22118 C0SUF4 11057969 Ki = 1200 nM T22118 CFJG64 11059058 IC50 = 7580 nM T22118 CE3J0B 11068912 Ki = 1200 nM T22118 CXP12A 11133602 Ki = 1100 nM T22118 CWC6E8 11152302 Ki > 1000 nM T22118 C3Q9UG 11154178 Ki = 0.2 nM T22118 CAY3B5 11175544 Ki > 1000 nM T22118 C0W4SM 11186523 Ki = 22 nM T22118 CN06GJ 11186895 Ki = 199 nM T22118 C9CTH8 11188446 Ki > 1000 nM T22118 CPX23W 11209208 IC50 > 10000 nM T22118 C6RXG7 11222979 Ki > 1000 nM T22118 C8RJ3D 11223303 Ki = 1.5 nM T22118 CF42AW 11233507 Ki > 1000 nM T22118 CKX06B 11235174 Ki = 0.5 nM T22118 CU8HM2 11268785 Ki > 1000 nM T22118 CM72YX 11269330 Ki = 0.3 nM T22118 C27GXZ 11277680 IC50 > 10000 nM T22118 CUJ2R7 11280344 Ki > 10000 nM T22118 C8J3QH 11282465 Ki = 443 nM T22118 C57GTA 11299968 IC50 > 10000 nM T22118 C1PDJ5 11306892 Ki = 7.1 nM T22118 CUXZ91 11311148 IC50 > 10000 nM T22118 C2GZD3 11311204 IC50 > 10000 nM T22118 CSA7U3 11313751 Ki > 1000 nM T22118 C5K8SP 11314647 Ki > 1000 nM T22118 CU82GC 11315254 Ki > 1000 nM T22118 C85FPO 11315462 Ki = 2.3 nM T22118 CJ2TH8 11326248 Ki > 1000 nM T22118 CSR03X 11326600 Ki > 1000 nM T22118 C0NRE8 11346967 Ki = 1651 nM T22118 CPA4W3 11349297 Ki = 405 nM T22118 C4XC2F 11349635 Ki > 1000 nM T22118 CCY23Q 11351639 Ki = 1730 nM T22118 CXWH42 11358377 Ki = 4748 nM T22118 CY24NV 11374299 Ki = 0.5 nM T22118 COD89G 11383046 Ki > 1000 nM T22118 CPQU06 11393136 Ki > 1000 nM T22118 CFN86P 11394557 Ki > 1000 nM T22118 C1V4EQ 11404156 Ki = 1676 nM T22118 CT32OJ 11406143 Ki = 1480 nM T22118 C3OL9U 11406615 Ki = 446 nM T22118 CGN10L 11408148 Ki = 1460 nM T22118 CV1AT8 11417923 Ki > 1000 nM T22118 CLH0N1 11429008 Ki > 1000 nM T22118 C85LYP 11430418 IC50 > 1000 nM T22118 CBN91Q 11439190 Ki = 2.8 nM T22118 C86CJB 11451022 Ki > 10000 nM T22118 CF6AM3 11451082 Ki > 1000 nM T22118 C0TKD2 11452896 Ki > 1000 nM T22118 CB3P6S 11452916 Ki = 0.7 nM T22118 C8L6ZI 11472028 Ki = 2621 nM T22118 C3MJK9 11474718 Ki > 1000 nM T22118 CK39HZ 11486421 Ki = 1.4 nM T22118 CYZ79A 11486571 Ki > 1000 nM T22118 CQL8F0 11487016 Ki > 1000 nM T22118 CTU1Z7 11488247 Ki = 0.6 nM T22118 CKV25P 11493746 Ki = 3.2 nM T22118 CR1HO4 11500181 Ki > 10000 nM T22118 CAU1R7 11500677 Ki = 82 nM T22118 CN63TR 11504230 Ki = 490 nM T22118 C16TWK 11508052 IC50 > 10000 nM T22118 CXWO08 11522273 IC50 > 10000 nM T22118 CQ5IN9 11522339 Ki = 8.7 nM T22118 CC6U7R 11522476 Ki = 509 nM T22118 C38QFE 11530118 IC50 > 10000 nM T22118 C75YUO 11536580 Ki > 10000 nM T22118 C2JT3I 11536995 Ki = 7.6 nM T22118 CQ08DH 11539632 IC50 = 7.5 nM T22118 CN3W7S 11543350 Ki > 10000 nM T22118 C8X0EM 11543992 Ki > 10000 nM T22118 C0AN1Y 11551474 Ki > 10000 nM T22118 C9VC7O 11551780 IC50 > 10000 nM T22118 C7S2WZ 11558055 Ki = 0.3548 nM T22118 CM8G3B 11558247 Ki = 9.3 nM T22118 C4HDA6 11558324 Ki > 10000 nM T22118 C1V5CH 11559090 Ki = 1810 nM T22118 C8GK0U 11566745 Ki = 20.7 nM T22118 CP8MF4 11573628 Ki = 3.1 nM T22118 C1TBC8 11573806 Ki = 9.4 nM T22118 C8NMI4 11575479 Ki = 120 nM T22118 C6JC2T 11580039 IC50 > 10000 nM T22118 C1M2CP 11589069 Ki = 2400 nM T22118 CU45DK 11595209 Ki > 10000 nM T22118 C5Q8XM 11595240 Ki = 0.46 nM T22118 CFC25K 11601627 Ki > 10000 nM T22118 C9D7OU 11616435 Ki > 10000 nM T22118 CN1P4I 11623343 Ki = 2 nM T22118 CIZ53S 11623652 Ki > 10000 nM T22118 CS4CR7 11631304 Ki = 767 nM T22118 CMX4K8 11633643 Ki > 10000 nM T22118 CG1C3D 11637457 Ki = 4 nM T22118 C2OU7Y 11638332 Ki > 10000 nM T22118 C35WZF 11639064 Ki = 755 nM T22118 CLZQ65 11644613 Ki > 10000 nM T22118 CHIW07 11652965 Ki > 10000 nM T22118 C1HDM5 11653679 Ki = 162.7 nM T22118 CO69ZI 11666419 Ki > 10000 nM T22118 CE34SW 11668495 Ki > 10000 nM T22118 CI26JH 11674133 Ki > 10000 nM T22118 CTK8R9 11678172 Ki = 970 nM T22118 CSQ4B1 11681599 Ki = 0.46 nM T22118 C06BEA 11694873 Ki > 10000 nM T22118 CRO95K 11695189 Ki > 10000 nM T22118 CN1SJ8 11696598 Ki > 10000 nM T22118 CKT7L2 11698732 Ki = 544.4 nM T22118 CB4H2O 11699469 Ki = 780 nM T22118 CDLW51 11701907 Ki > 10000 nM T22118 CJL61W 11706497 Ki = 2800 nM T22118 C0G1WQ 11709500 Ki > 10000 nM T22118 CI3N1K 11716230 Ki > 10000 nM T22118 CZ6NB8 11716438 Ki = 2.6 nM T22118 CZ7SJ2 11716449 Ki = 16.4 nM T22118 C9FTL5 11718008 Ki = 25.3 nM T22118 CGO56C 11720302 Ki = 570 nM T22118 C7PVL8 11730467 IC50 = 2750 nM T22118 C9X7MJ 11739647 Ki > 1000 nM T22118 C43XLH 11739648 Ki > 1000 nM T22118 CPG15O 11743399 IC50 > 1000 nM T22118 C2J7KO 11751611 Ki > 10000 nM T22118 CVJN50 11772639 Ki > 1000 nM T22118 C6T9RL 11773599 Ki > 1000 nM T22118 CV91RG 11778580 Ki = 3.2 nM T22118 CM82VH 11809382 Ki > 1000 nM T22118 CDX4W7 11957535 Ki = 0.17 nM T22118 CNXB23 11957706 Ki = 7 nM T22118 C8JQL7 11957735 IC50 > 10000 nM T22118 C7NV4W 12068769 Ki > 10000 nM T22118 CF4W7L 12269810 IC50 = 630 nM T22118 C4NWX9 12301195 Ki = 2116 nM T22118 CQIL96 12304090 Ki = 1189 nM T22118 CCLH20 12313091 Ki = 60 nM T22118 CWQ8M2 12442999 Ki = 135 nM T22118 C2CX7E 12668019 EC50 = 2 nM T22118 C3Y7TJ 12928470 Ki = 190 nM T22118 C6JX5B 12928483 Ki = 702 nM T22118 CCG14E 13091356 Ki > 10000 nM T22118 CYN95Z 13091359 Ki = 347 nM T22118 CC74ND 13373172 Ki = 136 nM T22118 CI5Y6N 13611248 Ki > 10000 nM T22118 C3W2EN 13697621 Ki = 1.2 nM T22118 CP2I9Z 13720692 Ki = 12 nM T22118 CN4Z2W 13851600 EC50 > 10000 nM T22118 CETG69 13864380 EC50 = 490 nM T22118 CA50UC 13864382 EC50 = 490 nM T22118 CWL63T 14021682 IC50 > 10000 nM T22118 C50HOI 14198585 Ki = 446.68 nM T22118 CIE29U 14198587 Ki = 26.92 nM T22118 CDE92A 14198590 Ki = 141.25 nM T22118 CNYA85 14198594 Ki = 281.84 nM T22118 COL2A4 14198597 Ki = 87.1 nM T22118 CTXB93 14198601 Ki = 177.83 nM T22118 CE1F9T 14371639 Ki = 7 nM T22118 CV08GM 14378574 Ki = 200 nM T22118 C4FLY3 14787971 Ki = 0.8 nM T22118 CEQG79 14787973 Ki = 0.4 nM T22118 C1TL0O 14787975 Ki = 1.6 nM T22118 CRD2I7 14787976 Ki = 531 nM T22118 C6R2OV 14787977 Ki = 513 nM T22118 CZVL61 14809027 EC50 = 2.1 nM T22118 C6ZUG1 15061351 IC50 = 1080 nM T22118 C3FKJ1 15111049 Ki = 4.1 nM T22118 C2UD7Q 15111050 Ki = 0.9 nM T22118 C3V8UK 15111051 Ki = 1.2 nM T22118 CO6ZI9 15111052 Ki = 48 nM T22118 CRE91W 15115512 Ki = 710 nM T22118 C4MD0E 15115513 Ki = 24000 nM T22118 CR57HC 15115514 Ki = 260 nM T22118 CLX2W5 15115515 Ki = 340 nM T22118 CK59LT 15115516 Ki = 3700 nM T22118 C8VT6W 15115519 Ki = 99 nM T22118 CV58UD 15115523 Ki = 2.3 nM T22118 CGC27M 15115524 Ki = 16 nM T22118 CHT4A5 15115525 Ki = 5.3 nM T22118 C1HAM3 15115530 Ki = 10000 nM T22118 CK46HZ 15225749 Ki = 280 nM T22118 CO8BJ0 15225750 Ki = 494 nM T22118 C01REV 15548770 Ki = 2200 nM T22118 CJ8D3W 15696481 EC50 = 142 nM T22118 C24WUI 15696482 EC50 = 232 nM T22118 CZY90M 15696487 EC50 = 68.7 nM T22118 CBXG85 15723715 Ki = 2100 nM T22118 C8UO1X 15981509 EC50 = 29 nM T22118 C0G2EO 16007117 Ki = 4 nM T22118 CWMC70 16090814 Ki = 2.042 nM T22118 CP09RQ 16090821 Ki = 158.49 nM T22118 C8Y5LU 16219951 EC50 = 0.3 nM T22118 CZ2IS9 16660294 Ki > 10000 nM T22118 CGX0D5 16665071 Ki = 2 nM T22118 C7KP5T 17755866 Ki = 13.9 nM T22118 CX7VE8 17755867 Ki = 2.667 nM T22118 CUW8S4 17755868 Ki = 83 nM T22118 C3KA6Z 17755875 Ki > 10000 nM T22118 C4N1LS 17755991 Ki = 291 nM T22118 C6BE2Y 17755992 Ki > 10000 nM T22118 C10UQJ 17755999 Ki = 28.18 nM T22118 C6WO9X 17756101 Ki = 18.5 nM T22118 CI9RW0 17756102 Ki = 23.5 nM T22118 CDPT42 17756110 Ki > 10000 nM T22118 C0XG9B 17756212 Ki = 137 nM T22118 C6JQ1K 17756213 Ki = 70 nM T22118 C61OBX 19881394 Ki > 10000 nM T22118 C5IHG3 19964406 Ki > 100000 nM T22118 CG5NT4 20035572 Ki > 10000 nM T22118 C7Y0HC 21302486 Ki = 110 nM T22118 C94BPG 21460314 Ki > 10000 nM T22118 C3T5HF 21509921 Ki > 10000 nM T22118 CFN81Q 21527771 Ki = 22 nM T22118 CH59WN 21533446 Ki = 27 nM T22118 CL5A2V 21554999 Ki > 10000 nM T22118 C61LUT 21555004 Ki > 10000 nM T22118 CAH39X 21564536 Ki > 10000 nM T22118 CVF4N8 21786101 EC50 = 25 nM T22118 CT7XG9 21830793 Ki > 10000 nM T22118 CXD3E6 23625925 Ki = 38.9 nM T22118 CDH38J 23992579 Ki > 10000 nM T22118 C4UQL5 24133757 EC50 = 1870 nM T22118 C58AMS 24829343 Ki = 3360 nM T22118 C1OFA6 24837531 IC50 = 6510 nM T22118 CY21RE 24841480 Ki = 5900 nM T22118 C2T5EW 24847750 Ki = 37.3 nM T22118 CUW23K 24854106 Ki = 1900 nM T22118 C2OM6C 24863698 Ki = 63.1 nM T22118 CKF9G6 24878061 EC50 = 1100 nM T22118 C69AYD 24900557 Ki = 42.66 nM T22118 C4IGH9 24936042 Ki = 2800 nM T22118 CI8NL3 25071384 Ki = 970 nM T22118 C6F5SU 25071385 Ki = 430 nM T22118 CL7TN4 25071691 Ki = 670 nM T22118 C75ZIC 25071692 Ki = 930 nM T22118 C49ZFU 25072002 Ki = 210 nM T22118 C8OBV4 25072633 Ki = 1100 nM T22118 CS1CI4 25072941 Ki = 1400 nM T22118 CBKG34 25093832 Ki = 710 nM T22118 C3W6DQ 25096873 IC50 > 1000 nM T22118 CJK06X 25110705 Ki = 4.88 nM T22118 CE72YO 25110706 Ki = 39 nM T22118 CM3X9B 25110707 Ki = 190 nM T22118 CTV61A 25110708 Ki = 56 nM T22118 CVIB80 25110709 Ki = 6.81 nM T22118 C2FY7C 25128757 Ki = 3000 nM T22118 C5NW4M 25129807 Ki = 1220 nM T22118 CAV81B 25130157 Ki = 3930 nM T22118 C67QCG 25132869 Ki = 1710 nM T22118 CL84YJ 25141534 Ki = 4630 nM T22118 C4FXR9 25141535 Ki > 10000 nM T22118 CKBJ53 25141536 Ki > 10000 nM T22118 C8OGB1 25141538 Ki = 5060 nM T22118 CX04LB 25142456 EC50 = 32 nM T22118 C78HME 25212275 Ki = 203 nM T22118 CE6Z9I 25212276 Ki = 203 nM T22118 C76ROY 25256815 Ki = 346.74 nM T22118 C7JZ2D 25256816 Ki = 2691.53 nM T22118 C6PL1Y 25256817 Ki = 1737.8 nM T22118 C4MRQ0 27842480 IC50 > 50000 nM T22118 CYU71X 36791366 Ki = 565 nM T22118 C15PLV 40152769 Ki = 6500 nM T22118 CAM63X 42618195 IC50 > 1000 nM T22118 C8K4UF 42618197 IC50 > 1000 nM T22118 C7BPK4 42625205 Ki = 990 nM T22118 CS8OZ6 42625207 Ki = 678 nM T22118 CJ2TA7 42625211 Ki = 4960 nM T22118 CQ37BN 42625290 Ki > 10000 nM T22118 CXB28J 42625293 Ki = 3690 nM T22118 CYM0J6 42625295 Ki > 10000 nM T22118 CD9RN1 42626103 Ki = 931 nM T22118 CTW8G4 42626171 Ki > 10000 nM T22118 C0P3JR 42626172 Ki > 10000 nM T22118 CZ19KX 42626240 Ki > 10000 nM T22118 CTL2I7 42626243 Ki > 10000 nM T22118 C98BKP 42626313 Ki > 10000 nM T22118 C1VR4S 42626315 Ki = 6650 nM T22118 CRQ91B 42626318 Ki > 10000 nM T22118 CTYZ17 42626380 Ki > 10000 nM T22118 C1JK6E 42626381 Ki > 10000 nM T22118 C2AV1K 44190762 IC50 = 1530 nM T22118 CVG6X1 44209472 Ki = 180 nM T22118 CD5AB7 44209480 Ki = 238 nM T22118 C2NIU8 44241577 Ki = 94 nM T22118 CMG0J7 44241581 Ki = 124 nM T22118 CFEI56 44267161 IC50 = 13803.84 nM T22118 CIZ5W7 44267181 IC50 = 34673.69 nM T22118 C79YQZ 44276404 EC50 = 320 nM T22118 CWG0B7 44276405 EC50 = 63 nM T22118 CWS4K2 44276412 EC50 = 23 nM T22118 CNT6P3 44276414 EC50 = 18 nM T22118 CJEB02 44276535 EC50 = 110 nM T22118 CGC3Z5 44276551 EC50 = 8.6 nM T22118 CHG9P5 44276552 EC50 = 8.8 nM T22118 CT6XU0 44276556 EC50 = 38 nM T22118 C95QZD 44276557 EC50 = 230 nM T22118 CTUC23 44276572 Ki = 390 nM T22118 CLH93D 44276651 EC50 = 120 nM T22118 CTC47W 44276652 EC50 = 180 nM T22118 CG0F7S 44282985 EC50 = 100 nM T22118 C1CD2E 44319915 EC50 = 650 nM T22118 CDY52A 44319976 EC50 = 6.4 nM T22118 C2EK5U 44319988 EC50 = 1740 nM T22118 CD8L6W 44320001 EC50 = 5.2 nM T22118 C42XTH 44320002 EC50 = 37.6 nM T22118 CP1TJ8 44320024 EC50 = 1.3 nM T22118 CNE68U 44320026 EC50 = 5.8 nM T22118 C5WB3L 44320050 EC50 = 3.1 nM T22118 CR7E3H 44320053 EC50 = 16.4 nM T22118 CO9PN8 44320061 EC50 = 2.02 nM T22118 C95MTC 44320076 EC50 = 34.4 nM T22118 CU6O2V 44320092 EC50 = 1.02 nM T22118 CLEM57 44320116 EC50 = 13.6 nM T22118 CRG47P 44320123 EC50 = 67 nM T22118 COW08A 44320129 EC50 = 6.3 nM T22118 C8I2DS 44320218 EC50 = 237 nM T22118 C6GXH5 44320256 EC50 = 100 nM T22118 C1UBS3 44320257 EC50 = 89 nM T22118 CT9YX2 44320267 EC50 = 24 nM T22118 C5BHP1 44320303 EC50 = 12.5 nM T22118 C3I8CM 44320304 EC50 = 2730 nM T22118 C8S7ZY 44320327 EC50 = 46.5 nM T22118 C9QU3D 44320328 EC50 = 124 nM T22118 C65MXL 44320357 EC50 = 3.5 nM T22118 C7Z3CW 44320378 EC50 = 6.7 nM T22118 CYP6M3 44331310 Ki = 20 nM T22118 CWKN28 44339794 IC50 > 1000 nM T22118 CD9ZS8 44342270 IC50 = 2740 nM T22118 CKL64H 44358192 Ki = 1350 nM T22118 CJ80OW 44360984 Ki = 2300 nM T22118 CS8K1A 44360992 Ki = 1200 nM T22118 C3NZ7B 44361021 Ki = 1500 nM T22118 C5XJD8 44366021 Ki = 28 nM T22118 C6BZS0 44393403 Ki = 900 nM T22118 C5XC2B 44401042 Ki = 250 nM T22118 CD56EA 44401105 Ki = 154 nM T22118 CW3PC2 44401106 Ki = 19 nM T22118 C9WH7P 44401164 Ki = 3 nM T22118 CXT84G 44401243 Ki = 83 nM T22118 C1B4QL 44403095 Ki > 10000 nM T22118 C1YL7Z 44403098 Ki > 10000 nM T22118 CFV98A 44403101 Ki > 10000 nM T22118 C6OY9S 44403102 Ki > 10000 nM T22118 CH4SX6 44403105 Ki > 10000 nM T22118 C12FIH 44403106 Ki > 10000 nM T22118 C4LKC1 44404394 Ki > 10000 nM T22118 C3EJ4G 44404396 Ki > 10000 nM T22118 CF4S3Y 44405965 Ki = 516 nM T22118 CT3Z8U 44405980 Ki = 8550 nM T22118 C0BI5F 44405985 Ki = 566.8 nM T22118 C4NC8M 44405995 Ki = 1040 nM T22118 C0R5VL 44406003 Ki = 388.7 nM T22118 CL5C9T 44406077 Ki = 271.6 nM T22118 CO2H3T 44406799 Ki > 10000 nM T22118 CI70SN 44406862 Ki > 10000 nM T22118 C0R6PK 44406863 Ki > 10000 nM T22118 CDA3R0 44406866 Ki > 10000 nM T22118 CU52FA 44406881 Ki > 10000 nM T22118 C0EXA1 44407083 IC50 > 10000 nM T22118 CZ24HP 44408818 Ki = 22.91 nM T22118 CMW2Z8 44415338 Ki = 30 nM T22118 CQM07I 44415345 Ki = 47 nM T22118 C5O7LC 44415367 Ki = 154 nM T22118 C8YWJ4 44415368 Ki = 111 nM T22118 CX8TH3 44415382 Ki = 79 nM T22118 CS27IO 44415383 Ki = 56 nM T22118 CS6D0A 44415394 Ki = 103 nM T22118 CBQ71R 44415395 Ki = 150 nM T22118 CBYP84 44415450 Ki = 98 nM T22118 CO1L6U 44415473 Ki = 86 nM T22118 CQ13TC 44415490 Ki = 68 nM T22118 C35IJK 44415506 Ki = 3 nM T22118 CK50IL 44415507 Ki = 13 nM T22118 CQ57GR 44415517 Ki = 47 nM T22118 C4VWS0 44415518 Ki = 4 nM T22118 C8R3VX 44415535 Ki = 42 nM T22118 CZ0RO7 44415536 Ki = 3.6 nM T22118 C98EFJ 44415543 Ki = 157 nM T22118 C75DUR 44415544 Ki = 14 nM T22118 C6I8EF 44415551 Ki = 35 nM T22118 C3QAZ4 44415552 Ki = 7.7 nM T22118 C69NUI 44415558 Ki = 10 nM T22118 CC3YW8 44415559 Ki = 28 nM T22118 CDP0Y7 44415560 Ki = 51 nM T22118 C0MFJ2 44415567 Ki = 62 nM T22118 C58WLD 44415568 Ki = 148 nM T22118 CU2FG6 44415569 Ki = 1.6 nM T22118 C7RU3M 44415577 Ki = 22 nM T22118 CIR8U5 44415578 Ki = 11 nM T22118 CC2PQ3 44415579 Ki = 62 nM T22118 CD4CA5 44415582 Ki = 1232 nM T22118 CF90AU 44415584 Ki = 16 nM T22118 CDU6Y5 44415593 Ki = 3.8 nM T22118 C32GAH 44415594 Ki = 7.4 nM T22118 CWQ9G5 44415595 Ki = 7.8 nM T22118 C38COL 44415598 Ki = 65 nM T22118 COT4H5 44415599 Ki = 71 nM T22118 CUQ7W3 44415600 Ki = 60 nM T22118 CR89VA 44415601 Ki = 16 nM T22118 C3M4HU 44415605 Ki = 99 nM T22118 CFIT89 44415606 Ki = 86 nM T22118 CHQ92K 44415611 Ki = 15 nM T22118 C9U7DG 44415612 Ki = 65 nM T22118 C1TYG7 44415613 Ki = 237 nM T22118 CEO41K 44415615 Ki = 13 nM T22118 C8O5AW 44415622 Ki = 886 nM T22118 CW91OY 44415623 Ki = 571 nM T22118 CB9XC7 44415624 Ki = 22 nM T22118 CA3JN6 44415625 Ki = 156 nM T22118 CM5WN1 44415628 Ki = 14 nM T22118 CM2L3X 44415629 Ki = 9 nM T22118 CMT3S0 44415633 Ki = 11 nM T22118 C2I8XJ 44415638 Ki = 68 nM T22118 C64PWA 44415644 Ki = 1097 nM T22118 CIX23C 44415645 Ki = 238 nM T22118 C6PMV8 44415646 Ki = 4749 nM T22118 CCM42T 44415647 Ki = 2568 nM T22118 CVZH14 44415648 Ki = 83 nM T22118 C1MC3X 44415649 Ki = 20 nM T22118 C3GVI9 44415657 Ki = 10 nM T22118 C9NQ4B 44415658 Ki = 39 nM T22118 C4YT5G 44415670 Ki = 24 nM T22118 CH0BY5 44415672 Ki = 2.5 nM T22118 C1SQ8J 44415673 Ki = 28 nM T22118 CM84OB 44415685 Ki = 98 nM T22118 CY69CA 44415686 Ki = 130 nM T22118 CZ76OD 44415688 Ki = 12 nM T22118 CK59CO 44415689 Ki = 2.6 nM T22118 C7AZ5D 44415690 Ki = 3 nM T22118 CRJ9N4 44415701 Ki = 16 nM T22118 C0D4BL 44415702 Ki = 2 nM T22118 CAR0F2 44415703 Ki = 12 nM T22118 CEVY54 44415704 Ki = 3.2 nM T22118 C1MC6P 44415705 Ki = 7 nM T22118 C3KG7M 44415721 Ki = 12 nM T22118 C1XRF4 44415723 Ki = 3.4 nM T22118 C0R4OV 44415724 Ki = 4 nM T22118 CL4W5C 44415738 Ki = 175 nM T22118 CVS38E 44415743 Ki = 64 nM T22118 C8BU4E 44415745 Ki = 24 nM T22118 C3AWV2 44415758 Ki = 81 nM T22118 CH4O7P 44415759 Ki = 447 nM T22118 CK5C8A 44415786 Ki = 505 nM T22118 CQ5SV8 44415802 Ki = 56 nM T22118 CBMU18 44415804 Ki = 85 nM T22118 CK76UE 44415805 Ki = 294 nM T22118 C2S0MB 44415807 Ki = 48 nM T22118 C5EO4H 44415822 Ki = 49 nM T22118 CLY4R7 44415823 Ki = 86 nM T22118 CEP25B 44415824 Ki = 54 nM T22118 C95DPW 44415825 Ki = 503 nM T22118 CI5MF1 44415826 Ki = 7 nM T22118 C8JE2L 44415827 Ki = 6 nM T22118 CL0K9A 44415835 Ki = 31 nM T22118 C5ELF8 44415836 Ki = 26 nM T22118 CPE3D9 44415837 Ki = 191 nM T22118 C8D9WN 44415838 Ki = 51 nM T22118 C7IR4G 44415839 Ki = 47 nM T22118 C2V6LX 44415844 Ki = 23 nM T22118 C2KG8A 44415845 Ki = 88 nM T22118 C8I7FQ 44415848 Ki = 32 nM T22118 CMC2Z1 44415849 Ki = 44 nM T22118 CNUD41 44415954 Ki = 25.6 nM T22118 C89HPL 44417647 EC50 = 1100 nM T22118 CY0QJ2 44427970 Ki = 579 nM T22118 CBI86V 44439942 Ki = 0.82 nM T22118 C3HMI2 44439943 Ki = 0.56 nM T22118 C63PQV 44439944 Ki = 19 nM T22118 C2P4CI 44439945 Ki = 3.7 nM T22118 CZL97F 44455426 Ki = 899 nM T22118 C12XGE 44456400 Ki > 10000 nM T22118 C4DL5C 44469677 IC50 > 10000 nM T22118 CWPH50 44478261 Ki = 2520 nM T22118 C4SX7H 44537919 Ki = 551 nM T22118 CVD14L 44537925 Ki = 144 nM T22118 CRJ2I6 44554468 EC50 = 120 nM T22118 CX4D1K 44554470 EC50 > 10000 nM T22118 CYL5M9 44554472 EC50 = 150 nM T22118 C8F9OM 44554474 EC50 = 330 nM T22118 CLZ37T 44554643 EC50 > 10000 nM T22118 CV65YO 44554644 EC50 > 10000 nM T22118 CK2Y5P 44554649 EC50 = 230 nM T22118 C1MT5G 44554818 EC50 = 150 nM T22118 CQ1C7K 44554820 EC50 = 19 nM T22118 C7Z5IX 44554982 EC50 = 89 nM T22118 C7EI4P 44554984 EC50 = 210 nM T22118 CA3M1E 44554986 EC50 = 74 nM T22118 C7B4VN 44554987 EC50 = 400 nM T22118 CIZ2A5 44555137 EC50 = 360 nM T22118 CQ8JA9 44555138 EC50 = 3900 nM T22118 C16HEZ 44555445 Ki = 1264 nM T22118 CJSC58 44561317 Ki = 3.715 nM T22118 C9I2VT 44582113 Ki = 2041.74 nM T22118 C21GPX 44582115 Ki = 1778.28 nM T22118 CQEF30 44582140 Ki = 426.58 nM T22118 CVE23P 44582178 Ki = 281.84 nM T22118 COZ2M5 44582179 Ki = 8709.64 nM T22118 CS7P4T 44582187 Ki = 977.24 nM T22118 C6A8RM 44582461 Ki = 1698.24 nM T22118 C72BQU 44582489 Ki = 1737.8 nM T22118 CEM2D6 44582490 Ki = 1445.44 nM T22118 CLHG02 44582491 Ki = 2511.89 nM T22118 C1F6NA 44582517 Ki = 4897.79 nM T22118 CZK49H 44582518 Ki = 2398.83 nM T22118 CRCH48 44582675 Ki = 3828 nM T22118 CEJ4R8 44582676 Ki = 1410 nM T22118 C5QB4K 44582678 Ki = 1759 nM T22118 C01RCI 44582705 Ki = 1930 nM T22118 CPTZ81 44588898 Ki = 346 nM T22118 CC7M4H 44588932 Ki = 422 nM T22118 CP6ZA9 44591012 Ki = 879 nM T22118 CU37BO 44591098 Ki > 1000 nM T22118 CU48CL 44591099 Ki = 305 nM T22118 C7H9SE 44591134 Ki = 232 nM T22118 C6RLW0 44591135 Ki = 248 nM T22118 CJ89IW 45260733 Ki = 8.8 nM T22118 CG0BL7 45261538 Ki = 5 nM T22118 CYJ7P8 45379368 Ki > 10000 nM T22118 CU2CA7 45379369 Ki = 4.2 nM T22118 CT3K8Y 45379370 Ki = 28.5 nM T22118 CT3A1Q 45379373 Ki > 10000 nM T22118 C8TRE1 45379377 Ki = 1836 nM T22118 CML67J 45379515 Ki = 2101 nM T22118 C7MO3G 45481875 Ki = 501 nM T22118 CRL6D2 45481877 Ki = 963 nM T22118 C7S9HJ 45481888 Ki = 655 nM T22118 C0HPW1 45481889 Ki = 221 nM T22118 C47HZI 45481890 Ki = 492 nM T22118 C0CHF4 45482789 IC50 = 4900 nM T22118 CLO70J 45483261 Ki = 134.9 nM T22118 C7LD5K 45483269 Ki = 33.11 nM T22118 CI3WX2 46176232 Ki > 10000 nM T22118 C8YH5K 46180191 Ki > 10000 nM T22118 C5CET8 46180192 Ki > 10000 nM T22118 CEW06P 46180193 Ki > 10000 nM T22118 C9PBQ4 46180194 Ki > 10000 nM T22118 CP8RF4 46180256 Ki > 10000 nM T22118 CG8UK9 46180257 Ki > 10000 nM T22118 CO7SA6 46180258 Ki > 10000 nM T22118 CSY63N 46180259 Ki > 10000 nM T22118 C64TDV 46180261 Ki > 10000 nM T22118 CBM9O6 46180325 Ki > 10000 nM T22118 C1J3VH 46180327 Ki > 10000 nM T22118 CN3X9Q 46180328 Ki > 10000 nM T22118 C73KNC 46180331 Ki > 10000 nM T22118 CHN09F 46180394 Ki > 10000 nM T22118 CMS7T5 46180395 Ki > 10000 nM T22118 C62FUY 46180396 Ki > 10000 nM T22118 C10OKI 46180397 Ki > 10000 nM T22118 CM4R8A 46180398 Ki > 10000 nM T22118 CC7N8T 46180399 Ki > 10000 nM T22118 CSV1P2 46216855 Ki = 0.9 nM T22118 CY7NM6 46227242 Ki = 3019 nM T22118 CR9S7B 46227243 Ki > 10000 nM T22118 C9A8FV 46227273 Ki = 2349 nM T22118 CL3KU2 46227284 Ki = 1727 nM T22118 CS4O6A 46227317 Ki = 183 nM T22118 CE1L6H 46227320 Ki > 10000 nM T22118 CSQ9D5 46227325 Ki = 2070 nM T22118 CDI10H 46231541 Ki = 0.9 nM T22118 CMR89A 46231588 Ki = 0.5 nM T22118 CAW5U2 46231589 Ki = 2 nM T22118 CBGM85 46231645 Ki = 0.7 nM T22118 C9KI4E 46231646 Ki = 7 nM T22118 CYM51R 46231709 Ki = 0.7 nM T22118 C8SFI5 46231768 Ki = 2.8 nM T22118 C9BT2H 46231769 Ki = 5.7 nM T22118 CD6T5Y 46231770 Ki = 4.7 nM T22118 C3TIF9 46231771 Ki = 5.8 nM T22118 C0R6GH 46231772 Ki = 2.4 nM T22118 C1EW4S 46231782 Ki = 2.3 nM T22118 CF3NS8 46231783 Ki = 38 nM T22118 C6JM5T 46231784 Ki = 0.6 nM T22118 CFJP50 46231833 Ki = 2.3 nM T22118 CR9L3V 46231834 Ki = 152 nM T22118 C14XCV 46231835 Ki = 225 nM T22118 CD6IC3 46231845 Ki = 3 nM T22118 C38WBY 46231846 Ki = 2.6 nM T22118 C0A7GW 46231847 Ki = 2 nM T22118 CVT82S 46231848 Ki = 3.1 nM T22118 C9W1US 46231924 Ki = 4.4 nM T22118 CL7WX9 46231925 Ki = 1.8 nM T22118 CVG26Z 46231926 Ki = 0.2 nM T22118 CKJ09A 46231927 Ki = 1 nM T22118 CEMA94 46231992 Ki = 0.2 nM T22118 CLWO70 46231993 Ki = 0.4 nM T22118 C2BX8U 46231994 Ki = 0.6 nM T22118 C7FD2G 46231995 Ki = 0.6 nM T22118 C0IBN1 46232064 Ki = 2.3 nM T22118 CM0PC8 46232065 Ki = 0.9 nM T22118 CYV52A 46232066 Ki = 0.7 nM T22118 CT8X1D 46232067 Ki = 0.7 nM T22118 C8XW1L 46232134 Ki = 0.7 nM T22118 CCL53R 46232135 Ki = 0.6 nM T22118 C0WJ5L 46850462 Ki = 22000 nM T22118 CN3RH6 46850464 Ki = 22000 nM T22118 C03LTM 46869265 EC50 = 0.64 nM T22118 C6BD5G 46905072 Ki = 4900 nM T22118 C7FX8L 46931072 Ki = 620 nM T22118 CR40BA 49836386 IC50 = 7200 nM T22118 C0M5XC 49836496 IC50 = 25000 nM T22118 C6OQV2 49862237 Ki > 1000 nM T22118 C1G7IZ 49866139 EC50 = 4.3 nM T22118 C2RY0J 50878551 Ki > 10000 nM T22118 C1W6TV 50898777 Ki > 10000 nM T22118 CXMZ73 50898778 Ki > 10000 nM T22118 CE4KP1 51050257 Ki > 10000 nM T22118 C6XY8V 52938728 Ki = 2700 nM T22118 CY2SH8 52939845 Ki > 5000 nM T22118 C7U0IC 52939846 Ki > 5000 nM T22118 C3S7HN 52939977 Ki > 5000 nM T22118 CLK7J6 52939978 Ki > 5000 nM T22118 CA16IT 52939979 Ki > 5000 nM T22118 CZ37RM 52939980 Ki > 5000 nM T22118 C19ZKQ 52946556 Ki = 0.39 nM T22118 C5C8ZN 53317208 Ki = 1900 nM T22118 CSM53O 53317282 Ki = 1600 nM T22118 C8JO1K 53317511 Ki = 3700 nM T22118 CKXS49 53317727 Ki = 340 nM T22118 C36MWP 53318500 Ki = 2007 nM T22118 CA31DT 53318564 Ki = 910 nM T22118 CU4CR9 53318565 Ki = 1174 nM T22118 CM5N9H 53320353 Ki > 5000 nM T22118 C5DL8F 53321194 Ki = 1307 nM T22118 CZ5AN7 53322729 Ki > 5000 nM T22118 C0WT8G 53322769 Ki > 5000 nM T22118 C32YWL 53324045 Ki = 135 nM T22118 C35GJZ 53325137 Ki = 735 nM T22118 CRQF15 53325242 Ki = 798 nM T22118 CQ8I3D 53326670 Ki > 5000 nM T22118 C76BWN 53327662 Ki = 1300 nM T22118 CUCE20 53327664 Ki = 380 nM T22118 CC8J5W 53328718 Ki = 4200 nM T22118 CY85HJ 53328720 Ki = 141 nM T22118 C79AYQ 53328901 Ki = 150 nM T22118 CMV95A 53328903 Ki = 140 nM T22118 CLZ09P 53359025 Ki = 209 nM T22118 C47KPJ 53362716 Ki = 2400 nM T22118 CU7W2I 53362841 Ki = 4200 nM T22118 CT81QW 53494976 EC50 = 570 nM T22118 CNDU46 53494978 EC50 = 584 nM T22118 C2RBG9 53494980 EC50 = 438 nM T22118 CU3M5C 54585745 Ki > 10000 nM T22118 CL5I1R 54753271 Ki > 10000 nM T22118 CQ3AR0 56589560 Ki = 6.1 nM T22118 C4XGR3 56589561 Ki = 114 nM T22118 C9PHZ3 56594402 Ki > 10000 nM T22118 C82IVX 56594533 Ki = 640 nM T22118 CT4J5C 56594534 Ki = 10.3 nM T22118 CU0NE5 56672197 Ki > 10000 nM T22118 CB0P9N 56944383 Ki = 3.3 nM T22118 CL16UQ 56949326 IC50 < 10000 nM T22118 C1TC7Q 56963799 Ki > 10000 nM T22118 CDZU04 57335757 EC50 > 100000 nM T22118 CV08WY 57391216 Ki = 495 nM T22118 C07PMA 57391307 Ki = 135 nM T22118 CWT20M 57393083 Ki = 134 nM T22118 CD4A3P 57396484 Ki = 259 nM T22118 C3GW6L 57398351 Ki = 126 nM T22118 CZX05B 57401706 Ki = 265 nM T22118 CYN38R 57401819 Ki = 589 nM T22118 CO0XD2 57401820 Ki = 52 nM T22118 CX0B5M 57403525 Ki = 130 nM T22118 CLWD45 57459488 Ki >= 6200 nM T22118 C4MV2N 60149678 Ki > 100000 nM T22118 C2Q5VD 60165416 Ki = 1897 nM T22118 C5RUP6 60167166 Ki = 1273 nM T22118 CGF3J5 66572162 IC50 = 9650 nM T22118 C34GMW 69599704 Ki > 10000 nM T22118 CPU15Z 70682088 Ki = 23.76 nM T22118 C9VL7R 70682090 Ki = 337.7 nM T22118 C6EI2D 70684206 Ki = 64.12 nM T22118 CL4RH5 70684207 Ki = 1440.62 nM T22118 C6PD9Q 70684338 Ki > 100000 nM T22118 CTHV58 70684339 Ki > 100000 nM T22118 COY65E 70684965 Ki = 270 nM T22118 C7GB8C 70686343 Ki = 52.34 nM T22118 CB9V3R 70686493 Ki > 100000 nM T22118 C1P3GF 70686494 Ki > 100000 nM T22118 C3V5QJ 70686495 Ki = 7000 nM T22118 C2U6KV 70688594 Ki > 100000 nM T22118 CBD3K8 70690497 Ki = 182.41 nM T22118 CS9H5V 70690498 Ki = 7.97 nM T22118 CF7X1W 70690499 Ki = 35.79 nM T22118 C1K3XW 70690500 Ki = 2.5 nM T22118 CG80JF 70690651 Ki = 42000 nM T22118 CZH6F9 70690652 Ki = 8000 nM T22118 C6TJA5 70690653 Ki = 49000 nM T22118 C6O8GF 70692652 Ki = 106.45 nM T22118 C7ZMB3 70692653 Ki = 74.51 nM T22118 C9J3TO 70692655 Ki = 17.29 nM T22118 C96FHP 70692656 Ki = 28.9 nM T22118 CU82LJ 70692801 Ki = 40800 nM T22118 C18ETD 70692802 Ki > 100000 nM T22118 C98YAU 70696888 Ki = 44000 nM T22118 CGXQ60 71041800 IC50 = 5750 nM T22118 C3J4SN 71041846 IC50 > 10000 nM T22118 CBF6Z8 71109804 Ki = 7.5 nM T22118 C5U4XV 71109897 Ki = 4.2 nM T22118 CC43QK 71151588 Ki > 1000 nM T22118 C2AQ7H 71195187 Ki > 1000 nM T22118 CON49H 71261649 Ki = 6.6 nM T22118 CSC3R7 71450213 Ki > 10000 nM T22118 C9VZ8J 71450550 Ki = 2979 nM T22118 CDI84E 71450922 IC50 > 10000 nM T22118 CYOA05 71451380 Ki = 0.94 nM T22118 C08KHB 71452040 Ki > 10000 nM T22118 C0XW8E 71452041 Ki > 10000 nM T22118 C43IWS 71453989 IC50 = 1100 nM T22118 CQMK12 71454927 Ki = 550 nM T22118 CDSX56 71457372 Ki > 10000 nM T22118 C3L2SU 71461395 Ki >= 6200 nM T22118 C9VE0P 71462090 Ki = 921 nM T22118 CQ2N0J 71508866 IC50 > 10000 nM T22118 C2K3CV 71524613 Ki > 5000 nM T22118 CE92DF 71528209 Ki = 12513 nM T22118 CWQ5R6 71562963 Ki = 244 nM T22118 CG1ZU7 71562964 Ki = 4 nM T22118 CI3EW5 71562965 Ki = 3340 nM T22118 C51IHJ 71562966 Ki = 252 nM T22118 CW2V1F 71563082 Ki = 45.9 nM T22118 C4ZKF0 71563083 Ki = 5.5 nM T22118 CR8UF1 71563084 Ki = 2 nM T22118 C50YDS 71716758 IC50 > 10000 nM T22118 CGU06V 71717958 IC50 > 10000 nM T22118 CW35XI 71722291 EC50 = 316 nM T22118 C4EC8K 71722293 EC50 = 21.9 nM T22118 C4FJV9 71722295 EC50 = 78 nM T22118 C8H5OT 71722297 EC50 = 117 nM T22118 C3SDV1 71722299 EC50 = 10.5 nM T22118 CY4NH1 71722300 Ki = 135 nM T22118 CQO30I 71733932 Ki = 18000 nM T22118 C93QMB 71733935 Ki = 13000 nM T22118 C31THM 72164180 Ki > 10000 nM T22118 C56VLM 72164181 Ki > 10000 nM T22118 CD8A9K 72164182 Ki = 2541 nM T22118 C4C0BH 72164183 Ki > 10000 nM T22118 CQU81Y 72164299 Ki > 10000 nM T22118 CF0H7K 72164300 Ki > 10000 nM T22118 C7WM5U 72164301 Ki > 10000 nM T22118 C4HO2U 72164302 Ki > 10000 nM T22118 CWH6T3 72548703 IC50 = 0.21 nM T22118 CIR7G1 72699716 Ki = 128.14 nM T22118 C9Y3DG 72699717 Ki = 133.05 nM T22118 CRMC07 72699718 Ki = 379.28 nM T22118 C4X9AO 72699812 Ki = 26.33 nM T22118 C5K9JW 72699815 Ki = 16.43 nM T22118 CZV6D5 72699816 Ki = 61.75 nM T22118 CIDS43 72699817 Ki = 62.19 nM T22118 C6J8GM 72699818 Ki = 66.21 nM T22118 CC8PL5 72699903 Ki = 45.82 nM T22118 C7YTK9 72699904 Ki = 718.74 nM T22118 CC65OA 73213195 Ki > 10000 nM T22118 CW83DK 73213196 Ki > 10000 nM T22118 CCV91B 73346042 Ki > 10000 nM T22118 CVA1D2 74223726 Ki = 113 nM T22118 CYRZ81 75201899 EC50 = 10 nM T22118 C2E7QW 75201901 EC50 = 0.2455 nM T22118 CO1Z7Q 75201961 EC50 = 1.175 nM T22118 CJG57Z 75202022 EC50 = 0.3 nM T22118 C8IDL3 75306277 Ki = 25.12 nM T22118 CZFW19 76314267 Ki = 30199.52 nM T22118 CIB40D 76321554 Ki = 8128.31 nM T22118 CS9F1X 76321556 Ki = 3890.45 nM T22118 C97LOB 76325150 Ki = 3890.45 nM T22118 CCR29U 76325152 Ki = 6606.93 nM T22118 C6GBK1 76325154 Ki = 1148.15 nM T22118 CLP59V 76325156 Ki = 10471.29 nM T22118 C2O0FW 76328713 Ki = 416.87 nM T22118 CZFD79 76335466 EC50 = 83 nM T22118 C28RIZ 76518514 Ki > 10000 nM T22118 CWI52H 77974401 Ki = 583 nM T22118 CS0DG1 85470885 EC50 = 460 nM T22118 C8EWX5 85658088 Ki = 861 nM T22118 CJ9K3T 86290953 EC50 = 1.11 nM T22118 C68RGH 86293768 EC50 = 3.66 nM T22118 CT6U8D 86302251 EC50 = 440 nM T22118 CM6X4U 86764103 EC50 = 5.3 nM T22118 CU84PK 90134199 EC50 = 12 nM T22118 CUKL15 90134211 EC50 = 21.88 nM T22118 C7J9VM 90134269 EC50 = 10 nM T22118 CW2TU5 90134304 EC50 = 153 nM T22118 CHV29I 90142280 Ki = 121 nM T22118 C80SXV 90644057 Ki = 2344 nM T22118 C20EPB 90644058 Ki = 641 nM T22118 C04MRN 90644059 Ki = 389.05 nM T22118 CIA8J4 90644060 Ki = 837 nM T22118 CY8TP0 90644061 Ki = 260 nM T22118 CKV24H 90644062 Ki = 222 nM T22118 CW2ZC4 90644063 Ki = 521 nM T22118 CLG60I 90644064 Ki = 7939 nM T22118 CKLN72 90644065 Ki = 1172 nM T22118 C7G5VH 90644066 Ki = 1408 nM T22118 CDPE48 90644071 Ki = 274 nM T22118 CLFV10 90644226 Ki = 150 nM T22118 CZ7LD8 90644227 Ki = 240 nM T22118 C35GPQ 90644228 Ki = 180 nM T22118 CZI30L 90644230 Ki = 3500 nM T22118 CACG19 90666899 Ki = 33.88 nM T22118 CODM50 90666903 Ki = 36.31 nM T22118 CNB56Y 90899701 IC50 = 390 nM T22118 CQR04O 92044504 EC50 = 0.87 nM T22118 CCV0I4 92640710 Ki > 100000 nM T22118 COA3U6 102262219 Ki = 11000 nM T22118 C1N5WJ 117720272 EC50 = 5.8 nM T22118 CIK45N 117949627 Ki = 86.98 nM T22118 CSH7K4 117949705 Ki = 77 nM T22118 C47STN 118445551 Ki = 98.9 nM T22118 CD4S9R 118709751 Ki = 4093 nM T22118 CO8E9F 118711252 Ki = 334 nM T22118 CJY9D7 118711253 Ki = 351 nM T22118 CFJE45 118711254 Ki = 665 nM T22118 CK1A2W 118711255 Ki = 277 nM T22118 CNQJ96 118711256 Ki = 370 nM T22118 CJ91QY 118711257 Ki = 292 nM T22118 C42YEC 118711258 Ki = 756 nM T22118 CU6BT0 118711259 Ki > 1000 nM T22118 C97RTC 118711260 Ki > 1000 nM T22118 CM47VI 118711261 Ki > 1000 nM T22118 CX3M2Z 118711262 Ki = 216 nM T22118 CN59OU 118711263 Ki = 912 nM T22118 CXI0S9 118711264 Ki > 1000 nM T22118 CW3F4T 118711265 Ki = 349 nM T22118 C4UAV9 118711266 Ki > 1000 nM T22118 C83MBF 118711267 Ki > 1000 nM T22118 C9FH2L 118711268 Ki > 1000 nM T22118 CBP47E 118711269 Ki > 1000 nM T22118 C7W2QM 118711270 Ki > 1000 nM T22118 C6QS7R 118711271 Ki > 1000 nM T22118 C6ZF8M 118711272 Ki > 1000 nM T22118 CDP7I9 118711273 Ki > 1000 nM T22118 CAF7I0 118711274 Ki > 1000 nM T22118 CUV5Y0 118715454 EC50 > 30000 nM T22118 CK98PG 118717796 Ki = 403.42 nM T22118 C43TKI 118717797 Ki = 633.79 nM T22118 CYW82N 118721287 Ki > 1000 nM T22118 CD21PC 118731187 IC50 = 6000 nM T22118 CW68KD 121304458 Ki > 100000 nM T22118 C35WTP 122177641 Ki = 2600 nM T22118 C8OS7B 122177642 Ki = 3900 nM T22118 CV2AT4 122177644 Ki = 23000 nM T22118 CB16GY 122177645 Ki = 2900 nM T22118 CH9SX5 122180956 Ki = 2600 nM T22118 CCV9D5 122181326 Ki = 1300 nM T22118 C5D1NC 122181329 Ki = 1300 nM T22118 C05RGV 122181330 Ki = 3300 nM T22118 C3XGN0 122181333 Ki = 2200 nM T22118 CK5BP3 122189387 Ki = 1700 nM T22118 C8JV3W 122189388 Ki = 210 nM T22118 CV1U4Q 122189389 Ki = 1500 nM T22118 C4PBA3 122189390 Ki = 160 nM T22118 CD7UN3 122189391 Ki = 620 nM T22118 C14FCX 122189392 Ki = 120 nM T22118 C1NIK8 122189393 Ki = 110 nM T22118 C9KXH4 122189394 Ki = 110 nM T22118 CVJ3R4 122191605 Ki = 480 nM T22118 C2J4ZX 122191607 Ki = 250 nM T22118 C7ODW3 122195524 Ki > 900 nM T22118 C71KZQ 122205437 Ki = 60 nM T22118 C30ZRC 122205438 Ki = 40 nM T22118 CM57GR 126720252 Ki = 7600 nM T22118 C09YOS 127027905 Ki > 10000 nM T22118 CE9MN1 127028185 Ki > 10000 nM T22118 C9SC6E 127028505 Ki > 10000 nM T22118 CJ4YC0 127031397 Ki = 19 nM T22118 CBU9G2 127031398 Ki = 40 nM T22118 CE1IA7 127031399 Ki = 6.7 nM T22118 C4WKG9 127031403 Ki = 12 nM T22118 CEDM28 127031404 Ki = 833 nM T22118 CV5UH0 127031405 Ki > 10000 nM T22118 CHN9X2 127031422 Ki = 12.4 nM T22118 C0CY9W 127031423 Ki = 7.8 nM T22118 CNH2V8 127031424 Ki = 11 nM T22118 C2W0HL 127031949 Ki = 3111 nM T22118 CZ61LK 127034966 IC50 > 5011.87 nM T22118 CA0SN5 127034967 EC50 > 5011.87 nM T22118 CQ0ZT9 127035062 Ki = 1682 nM T22118 CO53TS 127035828 Ki > 1000 nM T22118 CY7LP9 127035829 Ki > 1000 nM T22118 CR29BS 127035830 Ki > 1000 nM T22118 CU9C4S 127041952 Ki > 100000 nM T22118 C35GAL 127045853 Ki = 4500 nM T22118 C17LBT 127045854 Ki = 2800 nM T22118 CJ8GS7 127045855 Ki = 890 nM T22118 C2E1ZA 127046948 Ki = 6800 nM T22118 CTI5Z8 127046949 Ki = 2800 nM T22118 C4D6BQ 127046950 Ki = 430 nM T22118 CM4CQ7 127046951 Ki = 2900 nM T22118 C29ERQ 127046952 Ki = 860 nM T22118 C78IFA 127047221 Ki = 430 nM T22118 CZL0U7 127047859 Ki = 960 nM T22118 CZ6XL5 127047996 Ki = 210 nM T22118 C3WIA6 129103318 IC50 = 366 nM T22118 CZ25ED 130442471 EC50 = 12.88 nM T22118 CF7EK5 130442473 EC50 = 2.692 nM T22118 C50GOC 130442480 EC50 = 1.7 nM T22118 C4PZ0M 130442508 EC50 = 75.86 nM T22118 C2ST3W 130442514 Ki = 6.8 nM T22118 CYC76M 130442534 Ki = 8.5 nM T22118 C04UTE 130442557 Ki = 376 nM T22118 C5XK7A 130442561 Ki = 56.3 nM T22118 CM04RF 130442572 EC50 = 2.291 nM T22118 CRU8J0 130442590 EC50 = 5.754 nM T22118 C9DBU8 132016545 EC50 = 165 nM T22118 CY8B9L 132060743 Ki = 1804 nM T22118 CAVB41 132584404 Ki > 10000 nM T22118 CJ6C3E 134135947 Ki = 2.3 nM T22118 CSM98N 134137323 Ki = 9.7 nM T22118 C5RTN3 134139606 Ki = 1.3 nM T22118 CJE86B 134143833 Ki = 12 nM T22118 C0J1IR 134145434 Ki = 4.2 nM T22118 CB0NS6 134147903 Ki = 31 nM T22118 CJ5W4V 134149077 Ki = 65 nM T22118 CBU81N 134149168 Ki > 10000 nM T22118 CUFG17 134150400 Ki = 77 nM T22118 C5DX6R 134150645 Ki = 68 nM T22118 C2MAK7 134150852 Ki = 32 nM T22118 CW7AH9 134151737 Ki = 11 nM T22118 C8BI7V 134151764 Ki = 2.2 nM T22118 CW5VZ9 134155502 Ki = 5.3 nM T22118 C08MHZ 134157446 Ki = 7.7 nM T22118 C1GY2T 135156251 EC50 > 10000 nM T22118 C5OU1T 135409492 Ki = 395 nM T22118 CQ0SY6 135458464 Ki = 3799 nM T22118 C4PM9W 135515431 Ki = 66 nM T22118 C5KE3N 135986088 Ki = 866 nM T22118 C4GLA0 136043854 Ki = 583 nM T22118 CS7ZU5 136043855 Ki = 3106 nM T22118 CQC47B 136043856 Ki = 835 nM T22118 CF2BK1 136043857 Ki = 637 nM T22118 CP3XN7 136043859 Ki = 482 nM T22118 C89VLZ 136056636 Ki = 260 nM T22118 CN8BJ2 137632607 Ki = 8800 nM T22118 C3R2LO 137632761 Ki > 20000 nM T22118 C3PF9Z 137633454 Ki = 4000 nM T22118 COF9I6 137633705 Ki = 2900 nM T22118 C8YM6U 137633863 Ki = 1000 nM T22118 CN1I7A 137634153 Ki = 6000 nM T22118 C6FRJ5 137634397 Ki = 3800 nM T22118 CPHI76 137635364 Ki = 860 nM T22118 C8ZFQ6 137635685 Ki = 1100 nM T22118 CZ36LE 137636066 Ki = 2700 nM T22118 CAL1W4 137636298 Ki > 20000 nM T22118 CAQ6I5 137636351 Ki = 210 nM T22118 C6GWQ3 137636460 Ki = 1700 nM T22118 CQ20FO 137636498 Ki = 1500 nM T22118 CZU6N5 137636581 Ki = 5700 nM T22118 C0YDQ5 137637428 Ki = 7700 nM T22118 C49VDK 137638973 Ki = 600 nM T22118 C1HX3Z 137639304 Ki > 20000 nM T22118 CC16HE 137640152 Ki = 17000 nM T22118 CZP68A 137640189 Ki = 12000 nM T22118 CB2NO0 137640203 Ki = 410 nM T22118 CV49MZ 137640371 Ki = 1400 nM T22118 CCU7L3 137640391 Ki = 860 nM T22118 C8IO0R 137640836 Ki > 20000 nM T22118 C6PT7L 137642033 Ki > 20000 nM T22118 C94WSH 137642380 Ki = 240 nM T22118 CAC6W0 137643122 Ki > 20000 nM T22118 C71XIQ 137643132 Ki = 7500 nM T22118 CK51LB 137643309 Ki = 1300 nM T22118 C3O0FX 137643951 Ki = 1200 nM T22118 C34PUI 137644833 Ki = 470 nM T22118 CVX6T1 137644966 Ki = 250 nM T22118 C4PV8U 137645196 Ki > 20000 nM T22118 CNH95X 137645574 Ki = 5400 nM T22118 C3TP2G 137645830 Ki = 5300 nM T22118 CYH5U9 137647533 Ki > 20000 nM T22118 CR3Z6M 137651073 Ki = 280 nM T22118 CW4T6D 137651322 Ki = 12000 nM T22118 C15YDU 137651936 Ki = 800 nM T22118 CX30HQ 137653096 Ki > 15000 nM T22118 C4C6EV 137653986 Ki > 20000 nM T22118 COTX19 137654511 Ki > 20000 nM T22118 CF5Y2A 137654675 Ki = 4700 nM T22118 CLI4D8 137655029 Ki = 11000 nM T22118 C7RW9H 137655451 Ki = 3700 nM T22118 CJAZ13 137655556 Ki = 13000 nM T22118 C6CA5H 137655594 Ki > 20000 nM T22118 CDAN02 137655735 Ki = 900 nM T22118 CD16SQ 137655795 Ki = 4500 nM T22118 CA7F5N 137657115 Ki = 440 nM T22118 CV2CR4 137657153 Ki = 8600 nM T22118 CE0Y7P 137657322 Ki > 15000 nM T22118 CRT86S 137657427 Ki = 11000 nM T22118 CH76FP 137657951 Ki > 20000 nM T22118 CEZ07P 137659303 Ki = 920 nM T22118 CP9AN6 137659990 Ki = 1800 nM T22118 CP6US4 137660046 Ki = 2300 nM T22118 C5V4DQ 137660707 Ki > 20000 nM T22118 C42IDE 137660837 Ki = 2100 nM T22118 CNJ7D9 145867041 EC50 = 30 nM T22118 CJNG10 145966311 Ki = 610 nM T22118 CL58XS 145967572 Ki = 170 nM T22118 C58WSL 145967904 Ki = 1278 nM T22118 CB1FD8 145968810 Ki = 831 nM T22118 C48XNG 145969667 Ki = 174 nM T22118 CNZY06 145969934 Ki = 597 nM T22118 C61MSO 145970938 Ki = 542 nM T22118 CZF08O 145979741 Ki = 2242 nM T22118 C1XF0I 145979855 Ki = 1810 nM T22118 CO12QR 145979897 Ki = 1600 nM T22118 C87MSW 145980271 Ki = 10000 nM T22118 CUF6S4 145982261 Ki = 563 nM T22118 CP6DT9 145986441 Ki = 500 nM T22118 CNJH37 145986752 Ki = 10000 nM T22118 CO4LK7 145988180 Ki = 128 nM T22118 CUGO10 145988693 Ki = 300 nM T22118 CLWP79 145988779 Ki = 254 nM T22118 CLF26V 145990141 Ki = 680 nM T22118 CX0T9Y 145990190 Ki = 1680 nM T22118 CPW28Y 145990453 Ki = 800 nM T22118 C5OXL4 145992269 Ki = 2346 nM T22118 CRWE54 145993377 Ki = 800 nM T22118 CZ53LG 146025696 EC50 = 1000 nM T22118 CR6D1W 146025697 EC50 = 1300 nM T22118 CPYL02 146025698 EC50 > 10000 nM T22118 C9RO4I 146025699 EC50 = 602.56 nM T22118 C70ABE 146025700 EC50 = 54.95 nM T22118 C0YOF2 146025701 EC50 = 1.288 nM T22118 CRJD28 146025703 EC50 = 140 nM T22118 CO2M5D 146025704 EC50 = 15.49 nM T22118 CM79QY 146025705 EC50 = 88 nM T22118 CWCV47 146025706 EC50 = 35.48 nM T22118 CIQR27 146025707 EC50 = 100 nM T22118 C6O4YK 146025708 EC50 = 316.23 nM T22118 CX60SQ 146025709 EC50 = 1100 nM T22118 CT4FB0 146025710 EC50 = 61.66 nM T22118 CK89JR 146025711 EC50 = 79 nM T22118 C3A5OC 146025712 EC50 = 14.45 nM T22118 C2K3WN 146025713 EC50 = 0.2291 nM T22118 C9IC8Z 146025714 EC50 = 257.04 nM T22118 CO29GR 146025715 EC50 = 1.738 nM T22118 CJ4FN9 146025716 EC50 = 120 nM T22118 C78QIE 146025717 EC50 > 10000 nM T22118 CL2HP1 146025718 EC50 = 160 nM T22118 CGK05W 146025719 EC50 = 640 nM T22118 C35CWN 146025720 EC50 = 530 nM T22118 C6W7HL 146025721 EC50 = 109.65 nM T22118 CR94GO 146025724 EC50 = 190 nM T22118 CKY30W 146025725 EC50 = 770 nM T22118 C2LY5R 146025726 EC50 = 66.07 nM T22118 CC2G1V 146025727 EC50 = 2.188 nM T22118 CQX9D1 146025728 EC50 = 7.762 nM T22118 CXZ51B 146025729 EC50 = 180 nM T22118 C92EVC 146025730 EC50 = 269.15 nM T22118 C2JL8E 146025731 EC50 > 10000 nM T22118 CEY6N7 146025811 EC50 = 239.2 nM T22118 CZO92Q 146025812 IC50 = 100 nM T22118 CY97RS 146025813 EC50 = 150.2 nM T22118 C6NGR9 146025814 IC50 = 251.19 nM T22118 CXNT51 146025815 EC50 = 36.86 nM T22118 C7O0GT 146025816 EC50 = 246.8 nM T22118 CC1UL6 146025817 EC50 = 0.7943 nM T22118 C6IOM8 146025818 EC50 = 333.9 nM T22118 CT3I4V 146025819 EC50 = 194.3 nM T22118 CJ9I7W 146025820 EC50 = 14.45 nM T22118 CSL0Q5 146025821 EC50 = 0.38 nM T22118 CRJ3Z7 146025822 EC50 = 951.4 nM T22118 C9FY3J 146025823 EC50 = 41.36 nM T22118 CGTC03 146192950 EC50 = 127 nM T22118 CPU4B7 146192952 EC50 = 16.4 nM T22118 C68YPO 146192953 EC50 = 540 nM T22118 C3AH0G 146192955 EC50 = 81.2 nM T22118 CEW7M8 146192958 EC50 = 28 nM T22118 C5TY8P 146192959 EC50 = 112 nM T22118 CX4SD2 146192960 EC50 = 13.4 nM T22118 C2E0LC 146192964 EC50 = 287 nM T22118 C8XO4Z 146192966 EC50 = 172 nM T22118 C6P3SR 153287553 Ki > 10000 nM T22118 CV9G7Z 153287572 Ki > 10000 nM T22118 CO85KL 153287574 Ki > 10000 nM T22118 C5DQG2 155510939 IC50 > 10000 nM T22118 CQ83KZ 155512662 Ki > 10000 nM T22118 CHXY56 155513802 Ki = 1308 nM T22118 CL5G9Q 155513837 Ki = 1380 nM T22118 CH34RK 155514798 Ki = 1078 nM T22118 CUE5J3 155515907 Ki = 1758 nM T22118 CUM2N4 155515982 Ki = 200 nM T22118 CV12SD 155516041 Ki = 1349 nM T22118 CJ98ZK 155516236 Ki = 1668 nM T22118 C9ZAW0 155517266 Ki = 1711 nM T22118 CZ30CW 155518105 EC50 > 1000 nM T22118 C2UI6G 155519631 EC50 = 22 nM T22118 CUSA24 155519891 Ki > 10000 nM T22118 C8IYD1 155520455 Ki = 584.3 nM T22118 C5DSE0 155520996 Ki = 1148.2 nM T22118 CQBO46 155521159 EC50 = 410 nM T22118 CV7IG5 155522663 Ki > 5000 nM T22118 C8B2WR 155522744 IC50 > 10000 nM T22118 C2H3JL 155523073 Ki = 986 nM T22118 CQA76T 155523112 Ki = 992 nM T22118 C3E9DJ 155523127 Ki = 2906 nM T22118 CVQ68Y 155523770 Ki = 967 nM T22118 COH1Q5 155524191 Ki = 1288 nM T22118 CW7NT8 155524423 Ki = 891 nM T22118 CQX27T 155525357 Ki > 5000 nM T22118 CW65KS 155525705 Ki = 930 nM T22118 CK68PA 155526938 EC50 > 1000 nM T22118 CEN90X 155529453 Ki = 148 nM T22118 CKZ35G 155532475 Ki = 3631 nM T22118 C4LOR5 155532477 Ki = 1122 nM T22118 CQ12KS 155533996 Ki = 509 nM T22118 C8AX5N 155534186 Ki = 1423 nM T22118 CR7SF5 155534541 EC50 = 610 nM T22118 CHP2Z9 155535866 Ki = 649 nM T22118 CB79ZW 155536080 Ki > 10000 nM T22118 CY7XB4 155537335 EC50 = 360 nM T22118 CVFD68 155537516 Ki = 4898 nM T22118 CP0OJ4 155537850 EC50 > 1000 nM T22118 C13CSU 155537907 Ki = 636 nM T22118 C83KQL 155538443 IC50 = 1420 nM T22118 C3DIY2 155539246 Ki = 631 nM T22118 CPV48W 155539557 Ki = 794.3 nM T22118 C0D5ZP 155541775 EC50 = 210 nM T22118 CVK2M9 155543189 Ki = 940 nM T22118 C4ANI0 155543691 Ki = 2344 nM T22118 C08FTE 155544239 Ki = 1647 nM T22118 C7MCZ0 155546478 Ki = 871 nM T22118 CS6H3Z 155548298 EC50 = 18.3 nM T22118 C9E5LY 155549423 EC50 = 450 nM T22118 CN6I4P 155550431 Ki = 1457 nM T22118 C6N9PG 155550640 Ki = 992 nM T22118 CG7NR9 155550756 Ki = 832 nM T22118 C82QWR 155551173 Ki = 1981 nM T22118 CX8JA1 155552185 Ki = 360 nM T22118 C9T3AX 155552483 IC50 = 7420 nM T22118 CG70XQ 155552591 Ki = 1308 nM T22118 CB4F8Y 155552676 Ki = 368.7 nM T22118 CD5LC6 155554006 Ki = 818 nM T22118 C17XSQ 155555298 IC50 > 10000 nM T22118 CTP9I5 155558060 EC50 = 950 nM T22118 C36SYJ 155558844 Ki = 1084 nM T22118 C3U0RO 155560177 EC50 = 580 nM T22118 C7OZM6 155561446 Ki = 1047 nM T22118 CG3RL0 155561845 IC50 = 1030 nM T22118 CALB48 155561861 Ki > 10000 nM T22118 C2Z0HB 155562353 Ki = 1467.8 nM T22118 C0L1NB 155563581 EC50 > 1000 nM T22118 C0UN4V 155564747 Ki = 1509 nM T22118 CMH8I1 155565768 Ki = 1278 nM T22118 CK20WA 155566662 Ki = 1918 nM T22118 C6DPR8 155566974 Ki = 1122 nM T22118 C6HS0F 155567118 IC50 > 10000 nM T22118 C95RAP 155567835 Ki = 295.1 nM T22118 C5A6YM 155567869 Ki = 891 nM T22118 CV24CW 155568676 Ki = 1105 nM T22118 C73ERT 155568786 Ki = 1724.6 nM T22118 C42JKO 155569198 Ki = 1071 nM T22118 CH83UM 155569483 Ki = 5110 nM T22118 C3N9VU 10251906 Ki > 500 nM T22118 CP9TR0 10324985 Ki = 7396 nM T22118 CFMK68 3246545 Ki = 103 nM T22118 CB2VD8 44241743 Ki = 52 nM T22118 D00NQV 5041 Ki = 2830 nM T22118 D00SDJ 11237664 IC50 > 10000 nM T22118 D00YEB 25141414 Ki = 12 nM T22118 D01ADA 45269964 Ki = 278 nM T22118 D01ENR 2993172 Ki = 201 nM T22118 D01JXM 46222048 Ki > 1000 nM T22118 D01WWC 16573 Ki = 373 nM T22118 D02HNQ 46182736 IC50 > 10000 nM T22118 D02YCY 44568533 Ki = 78 nM T22118 D03JOX 11311147 IC50 > 10000 nM T22118 D03TPY 9885123 IC50 > 10000 nM T22118 D04AZE 3277600 Ki < 10000 nM T22118 D04TWX 9794475 IC50 > 10000 nM T22118 D05EQG 5265 Ki = 323 nM T22118 D05KUM 135446209 Ki = 203 nM T22118 D05QOF 14809026 EC50 = 8577 nM T22118 D05ZUX 44207909 Ki >= 1000 nM T22118 D06GGB 45271622 Ki = 31 nM T22118 D06LQH 167715 Ki = 1 nM T22118 D06QGD 11357862 IC50 > 10000 nM T22118 D06XKX 45269974 Ki = 669 nM T22118 D07CZJ 44447998 Ki = 23 nM T22118 D07IWZ 44568534 Ki = 2920 nM T22118 D07LRJ 5312149 Ki = 120 nM T22118 D07RYR 44396235 Ki = 379 nM T22118 D07ZOP 11470616 IC50 > 10000 nM T22118 D08TCX 11437461 Ki > 10000 nM T22118 D08UQU 24766199 Ki = 46 nM T22118 D09RPR 16737207 Ki > 10000 nM T22118 D09WBJ 10336538 Ki = 5500 nM T22118 D0B1GJ 44578927 Ki = 18 nM T22118 D0C5RZ 5610 Ki = 390000 nM T22118 D0D1PR 130907 Ki = 8.1 nM T22118 D0E1RX 11335419 Ki = 113 nM T22118 D0E3AL 56597938 Ki = 340 nM T22118 D0F0IA 11301655 Ki > 8000 nM T22118 D0FF6S 16038374 IC50 > 2000 nM T22118 D0G2CP 10404144 Ki = 12000 nM T22118 D0H2WQ 54562 Ki = 63 nM T22118 D0HG4U 11515697 Ki = 88 nM T22118 D0I2WQ 44579031 Ki = 31 nM T22118 D0I9KV 11220599 IC50 > 10000 nM T22118 D0J1HP 10378389 Ki = 6165.95 nM T22118 D0J3PJ 4331799 Ki = 1780 nM T22118 D0KX3X 44593524 Ki = 116 nM T22118 D0L3MJ 133538 EC50 = 0.2 nM T22118 D0L5MW 181743 Ki = 895 nM T22118 D0L7OM 6917970 Ki = 3.4 nM T22118 D0L8PI 5018 IC50 = 0.31 nM T22118 D0LR8X 1243 Ki = 0.3 nM T22118 D0M3PV 133633 Ki = 722 nM T22118 D0M5ZE 5311416 Ki < 10000 nM T22118 D0MT1N 45267373 Ki = 1340 nM T22118 D0NA2T 24800688 Ki > 5000 nM T22118 D0O7DA 37459 Ki = 2.3 nM T22118 D0P4BY 146265 Ki = 4.9 nM T22118 D0R8PL 44579030 Ki = 10 nM T22118 D0R8UU 44396220 Ki = 33.7 nM T22118 D0T1TU 68950 Ki = 1959 nM T22118 D0T2RY 9948320 Ki >= 1000 nM T22118 D0U6IL 13864381 EC50 = 490 nM T22118 D0V4FZ 173871 EC50 = 0.45 nM T22118 D0X8LG 11243002 IC50 > 10000 nM T13201 D00STL 644241 Ki = 29.3 nM T13201 D01MUR 68844 Ki = 3 nM T13201 D01WJL 4649 IC50 = 130000 nM T13201 D02FLB 516892 Ki = 12000000 nM T13201 D02PJA 24841 Ki = 300000 nM T13201 D02URS 4875 Ki = 300000 nM T13201 D02ZTJ 5339 IC50 = 3040 nM T13201 D03QGM 5355 Ki = 1200 nM T13201 D03RTS 2662 Ki > 10000 nM T13201 D03UOT 785 Ki = 10700 nM T13201 D04AIT 5280445 Ki > 10000 nM T13201 D04YZL 5234 Ki = 6000000 nM T13201 D05OFX 219078 Ki = 362 nM T13201 D05UYW 5284549 Ki = 500 nM T13201 D05VGL 11499245 Ki = 2015 nM T13201 D07HBX 338 Ki = 9900 nM T13201 D07INV 3295 IC50 = 15.71 nM T13201 D07MGA 72281 Ki > 10000 nM T13201 D07VDZ 5284627 Ki = 250 nM T13201 D08LFZ 3059 IC50 = 3380 nM T13201 D09NIA 2732 Ki = 348 nM T13201 D09VAZ 5565 Ki = 100000 nM T13201 D0A3HB 4943 Ki = 98900 nM T13201 D0AZ3C 5291 Ki = 31.9 nM T13201 D0AZ8C 5213 Ki = 1490 nM T13201 D0C2II 4100 Ki = 14 nM T13201 D0C8EU 5394 Ki > 50000 nM T13201 D0C8FX 3005837 Ki > 200000 nM T13201 D0E1SW 1986 Ki = 0.25 nM T13201 D0E9JM 4873 Ki = 6000000 nM T13201 D0GY5Z 2244 IC50 = 2710000 nM T13201 D0H8FH 3702 Ki = 51900 nM T13201 D0J4GO 3038 Ki = 25 nM T13201 D0J7RK 36811 Ki = 1920 nM T13201 D0K0OZ 5702160 Ki = 922.4 nM T13201 D0K1QD 3998 Ki = 25000 nM T13201 D0K8KX 5280343 Ki = 2680 nM T13201 D0L4JT 5333 Ki = 300 nM T13201 D0L6DA 119607 Ki > 50000 nM T13201 D0L7FM 4911 Ki > 10000 nM T13201 D0MA7C 23668193 Ki = 8400000 nM T13201 D0MD2L 129228 Ki > 10000 nM T13201 D0OT0O 44561 Ki = 24100000 nM T13201 D0PQ3G 3440 Ki = 62 nM T13201 D0R0FO 9823820 Ki > 10000 nM T13201 D0SH3I 387447 Ki = 1290 nM T13201 D0TG1H 3033 IC50 > 100000 nM T13201 D0U4UQ 3639 Ki = 328 nM T13201 D0U5QK 1983 Ki = 10000 nM T13201 D0V8QT 2708 Ki > 50000 nM T13201 D0VM2L 68740 IC50 > 10000 nM T13201 D0W5HK 216239 Ki > 10000 nM T13201 D0Y2IZ 5560 Ki = 345 nM T13201 D0Z3EI 6038 Ki = 6230 nM T13201 D0Z4UY 517045 Ki = 10800 nM T13201 D02JUW 460 Ki = 60200 nM T13201 D04IIU 216468 Ki = 30 nM T13201 D04PBH 5280804 Ki > 10000 nM T13201 D05NJI 5287541 Ki = 3450 nM T13201 D05ZXZ 491941 Ki = 323 nM T13201 D06DMQ 59472121 Ki > 50000 nM T13201 D06PII 5356 Ki = 374 nM T13201 D08BXT 1102 Ki = 1400 nM T13201 D09XQU 135413511 Ki > 50000 nM T13201 D0C2KF 11616111 Ki = 2200 nM T13201 D0I7IB 5222465 Ki = 511000 nM T13201 D0I7MT 5281807 Ki > 10000 nM T13201 D0L6HN 996 Ki = 10100 nM T13201 D0SC6I 517055 Ki = 730000 nM T13201 D0TO2R 30751 Ki > 10000 nM T13201 D0U3EP 445154 Ki = 2210 nM T13201 D0V0UK 82267 Ki = 0.31 nM T13201 D0W1SL 31404 Ki = 245200 nM T13201 D03SLR 445858 Ki = 2890 nM T13201 D08RPE 71607911 IC50 > 10000 nM T13201 D0F8XZ 19890 Ki > 100000 nM T13201 D0NH9P 135 Ki = 920 nM T13201 D0X2AU 23427 Ki > 100000 nM T13201 D07XPE 8249 Ki > 50000 nM T13201 D0LD9S 1103 Ki = 231000 nM T13201 CI0WH9 72 Ki = 1080 nM T13201 CJ28SX 127 Ki = 309000 nM T13201 CUT2V4 260 Ki = 4000000 nM T13201 COV5W3 402 Ki = 600 nM T13201 CSZ43B 540 Ki = 700 nM T13201 C97QXH 767 Ki = 12000000 nM T13201 C39CTO 768 Ki = 500 nM T13201 C1QDT0 781 Ki = 200000 nM T13201 CAD4R0 798 Ki = 27400 nM T13201 CW0R2L 944 Ki = 7000000 nM T13201 C6QX8I 1089 Ki = 118000000 nM T13201 CQV86E 1100 Ki = 18000000 nM T13201 C8W7BZ 1118 Ki = 18000000 nM T13201 CU12QE 1203 Ki = 2420 nM T13201 C6O0MZ 1491 Ki = 5200 nM T13201 CO4X7B 2456 Ki = 419 nM T13201 C5L7VX 2871 Ki = 61700 nM T13201 CQ0D8J 3469 Ki = 4200 nM T13201 CJ2F6P 5056 Ki = 2180 nM T13201 CTDR62 5235 Ki > 300000000 nM T13201 CKQC48 5238 Ki = 300000 nM T13201 CDJ4K6 5987 Ki = 0.021 nM T13201 C4V7LO 6738 IC50 = 3070000 nM T13201 CUP2F4 7043 Ki = 10400 nM T13201 C1CVT7 7121 Ki = 6830 nM T13201 CHG8L5 7322 IC50 = 420000 nM T13201 C6NC4O 7414 Ki = 10800 nM T13201 CJKY76 7420 Ki = 2370 nM T13201 C23KMD 7921 Ki = 4690 nM T13201 C6QYD8 8434 Ki = 7900 nM T13201 CD6O9A 8499 Ki = 3840 nM T13201 C46OQB 8697 Ki = 450000 nM T13201 C8VKM7 8929 Ki = 500 nM T13201 C40HCL 8987 Ki = 790000 nM T13201 CHP7I1 9016 Ki = 8210 nM T13201 CLYZ50 9338 Ki = 5700 nM T13201 CNM7L3 10199 Ki > 10000 nM T13201 CBIR94 10313 Ki = 83100 nM T13201 COU60V 10340 Ki = 15000000 nM T13201 CC30SK 10341 Ki = 13600 nM T13201 CM20CY 10393 Ki = 430000 nM T13201 C4NQE7 10787 Ki > 100000 nM T13201 CACI42 10953 Ki = 9600 nM T13201 C7H1FT 11335 Ki = 198300 nM T13201 CUG8B9 11418 Ki = 7560 nM T13201 CCPT31 11419 Ki = 8610 nM T13201 CV5PC3 11568 Ki = 4900 nM T13201 CL80QG 11820 Ki > 10000 nM T13201 CZLI84 12283 Ki = 57760 nM T13201 C14BYX 12662 Ki = 19100 nM T13201 CKA21F 14768 Ki = 570000 nM T13201 CUA0L6 14917 Ki > 300000000 nM T13201 CNI85U 15109 Ki = 9670 nM T13201 CQ4C5U 16523 Ki = 830 nM T13201 CS39YR 19654 Ki = 540000 nM T13201 CNGB21 20098 Ki = 690 nM T13201 C7OJ9Q 20125 Ki = 6480 nM T13201 C3LA1Z 20161 Ki = 7300 nM T13201 CMK0O4 20825 Ki > 10000 nM T13201 CF14KR 24247 Ki = 690000 nM T13201 CHW5M0 24268 Ki = 7000000 nM T13201 C4IZB8 24345 Ki = 95000000 nM T13201 CGR6D5 24413 Ki = 107000 nM T13201 C9M8EJ 24434 Ki = 7000000 nM T13201 CAN29U 24436 Ki = 63000000 nM T13201 C8S9AF 24445 Ki = 4790000 nM T13201 C3NG2U 24529 Ki = 8400000 nM T13201 CFM9L6 24530 Ki = 1200 nM T13201 CBT68I 24603 Ki = 790000 nM T13201 C3F1OY 25502 Ki = 570000 nM T13201 CE3U1F 26218 Ki = 540000 nM T13201 CF2XP3 26255 Ki > 200000000 nM T13201 CG04AY 26518 Ki > 100000 nM T13201 CDK20Z 27290 Ki > 50000 nM T13201 CWIZ67 28015 Ki = 600 nM T13201 C69RDT 32204 Ki = 8340 nM T13201 C7YZM4 33557 Ki = 1200 nM T13201 C4OU6D 35703 Ki = 31400 nM T13201 CY2GU3 60582 Ki = 249 nM T13201 C1N6SE 61127 Ki = 32145 nM T13201 CF26VS 61441 Ki = 370000 nM T13201 C6R1AJ 61609 Ki = 660000 nM T13201 CLMR98 61857 Ki = 13800000 nM T13201 CJ03HR 62481 Ki = 200000 nM T13201 CV28FU 62805 Ki > 10000 nM T13201 C5MJH8 64789 Ki > 50000 nM T13201 CN94KU 65008 Ki = 9310 nM T13201 C6DG9Q 65185 Ki = 14600000 nM T13201 C1NQ8E 65188 Ki = 21500 nM T13201 CT6YO0 66548 Ki = 7710 nM T13201 CCE63L 66634 IC50 = 1194 nM T13201 CMXS19 66814 Ki = 5354.1 nM T13201 CJ1Z2R 67125 Ki > 100000 nM T13201 C0ZK7U 67284 Ki = 5960 nM T13201 C8H4AT 67313 Ki = 170 nM T13201 CWXE69 67756 Ki = 12600 nM T13201 C26PTJ 67760 Ki = 13750 nM T13201 CJWD84 68154 Ki = 7970 nM T13201 CA3R7P 68351 Ki = 42 nM T13201 CB89AL 68982 Ki = 8700 nM T13201 CYEU83 69033 Ki = 18000 nM T13201 CVI38F 69809 Ki = 6640 nM T13201 CND3B8 70122 Ki = 316200 nM T13201 CX4HM3 70653 IC50 > 50000 nM T13201 C8U0VH 72597 Ki = 12.6 nM T13201 CJR96B 72879 Ki = 21000 nM T13201 CU79WI 74093 Ki = 6 nM T13201 CTMF08 75076 Ki = 770 nM T13201 C0I4UT 75077 Ki = 820 nM T13201 CE5RZ1 76509 Ki > 500000 nM T13201 C8DHG4 76792 Ki = 7840 nM T13201 CXG7Y0 76959 Ki = 4340 nM T13201 CVSE97 77456 Ki = 8800 nM T13201 C9V0ME 77547 Ki = 650 nM T13201 C6TS8J 77548 Ki = 710 nM T13201 CRXH06 77553 Ki > 10000 nM T13201 CZAX86 77578 Ki = 57800 nM T13201 C0PY5N 77754 Ki > 100 nM T13201 CX79KD 78297 Ki = 69.2 nM T13201 CX47BZ 78479 Ki = 115000 nM T13201 CCK8E1 79611 Ki = 35.7 nM T13201 C9QAS6 86986 Ki = 309000 nM T13201 C5BFK4 87432 Ki = 3660 nM T13201 CYIP60 89607 Ki = 7000 nM T13201 CM72DQ 90631 Ki = 910 nM T13201 CB5R7Y 92229 Ki = 3400 nM T13201 CB81UG 93577 Ki = 590 nM T13201 CJ01AO 94706 Ki = 50 nM T13201 C2GI9X 95801 IC50 > 50000 nM T13201 C40RWH 95840 Ki > 50000 nM T13201 C21JNS 95841 Ki > 10000 nM T13201 C1GQE3 97576 Ki = 6350 nM T13201 CEC01M 97598 Ki = 14730 nM T13201 CSGF32 99327 Ki = 315000 nM T13201 CA9YN2 99477 Ki > 10000 nM T13201 CV76MT 100187 Ki > 50000 nM T13201 CGM6A9 101263 Ki > 1000 nM T13201 C6K3MG 101424 Ki > 100000 nM T13201 C9Q4GE 102491 Ki = 4380 nM T13201 CI8DH1 103993 Ki > 10000 nM T13201 CD48YU 108326 Ki = 850 nM T13201 C27CDU 118534 Ki = 265000 nM T13201 CP4O2C 121255 Ki = 38000 nM T13201 CDP5M6 125623 Ki = 167 nM T13201 CN19UT 129695 Ki = 12300 nM T13201 CUX39B 132037 Ki = 12240 nM T13201 CCK5Y6 133125 Ki = 245 nM T13201 CVB67D 134560 Ki = 6 nM T13201 CD2HC7 138614 Ki = 7640 nM T13201 C2P0RH 139584 Ki = 110000 nM T13201 CUBQ92 145746 Ki = 38000 nM T13201 C9ZEP5 151399 Ki > 1000000 nM T13201 C47BCV 154989 Ki = 6490 nM T13201 CJ0FR9 155148 Ki = 9210 nM T13201 C50XVJ 159772 Ki = 630 nM T13201 C1SAJ0 162152 Ki = 310000 nM T13201 CW2Y7L 162287 Ki > 10000 nM T13201 CVH81Y 163571 Ki = 23000 nM T13201 C4U5KL 164000 IC50 = 290000 nM T13201 C8AO0Z 165323 Ki = 690 nM T13201 C6M0TK 167985 Ki = 500000 nM T13201 CU3WG6 179620 Ki = 9110 nM T13201 CE1VJ6 191826 Ki > 100000 nM T13201 CO96LR 192271 Ki = 28 nM T13201 C60KJD 192792 Ki = 163 nM T13201 C1N3AY 199210 Ki > 100000 nM T13201 C2GHM7 202375 IC50 > 50000 nM T13201 CSMP84 219987 Ki > 200000 nM T13201 C9K3VU 220023 IC50 > 50000 nM T13201 C90VSK 221131 Ki = 480 nM T13201 CEZU63 221227 Ki > 100000 nM T13201 C7DS2I 228958 Ki = 390 nM T13201 C2ED9N 236541 Ki > 10000 nM T13201 C14USE 239728 Ki > 50000 nM T13201 CW1E5G 239730 Ki > 50000 nM T13201 CP7Q8T 240910 Ki = 62000 nM T13201 CRP27E 245904 Ki = 14200 nM T13201 C6D1LY 246499 Ki = 30.2 nM T13201 C0B3OQ 253877 Ki = 4000000 nM T13201 C6DQU8 253881 Ki = 4000000 nM T13201 CLV79E 260228 Ki > 100000 nM T13201 CU45WA 260244 Ki > 100000 nM T13201 CI83OK 273360 Ki = 29620 nM T13201 C0UL5Y 276741 Ki = 155 nM T13201 CX3DK6 283995 Ki = 40000 nM T13201 C1QOB5 284045 Ki = 537311 nM T13201 C3QV5H 287064 Ki = 710 nM T13201 C26HNY 289493 Ki = 59200 nM T13201 C51UMX 294719 Ki = 6000 nM T13201 C83MLQ 295450 Ki > 50000 nM T13201 COE9A7 306924 Ki = 760 nM T13201 CAUO79 306968 Ki = 550 nM T13201 CM2N3X 307505 Ki = 158 nM T13201 C3W0AQ 307522 Ki = 92 nM T13201 C3WZI1 308397 Ki = 428 nM T13201 C6AKQ8 308411 Ki = 421 nM T13201 CL4GF1 308432 Ki = 442 nM T13201 C96DKW 310360 Ki = 5080 nM T13201 CY13EN 311156 Ki = 519 nM T13201 C12PJC 313721 IC50 > 50000 nM T13201 CQ67ZL 315810 Ki = 14250 nM T13201 COI7H8 317746 Ki = 87 nM T13201 CG3J6Q 323350 Ki = 31.2 nM T13201 CTX0Z3 327169 Ki = 72900 nM T13201 C8K5LE 338294 Ki > 10000 nM T13201 CXZ14S 341082 Ki > 50000 nM T13201 CP7X9H 342056 Ki > 10000 nM T13201 CMS5W4 343662 Ki > 10000 nM T13201 C5V2ZH 345312 Ki = 31 nM T13201 CH1C9B 351361 Ki = 147 nM T13201 COFX01 352863 Ki = 27000 nM T13201 CM9V8O 388547 Ki > 10000 nM T13201 CT3ZU4 388776 Ki = 136000 nM T13201 CH21KA 389641 Ki > 500000 nM T13201 C6CQO3 389642 Ki = 137000 nM T13201 CH0F9P 390929 Ki > 50000 nM T13201 CNPZ40 394897 Ki = 850 nM T13201 C4WC2P 394900 Ki = 900 nM T13201 CY39DK 394901 Ki = 460 nM T13201 CGUJ45 394902 Ki = 3 nM T13201 C2G6DI 394904 Ki = 5 nM T13201 C9NF6V 395814 Ki = 59800 nM T13201 CHU17A 395815 Ki = 10 nM T13201 C5TON3 395826 Ki = 3 nM T13201 CL5WQ3 396510 Ki = 8 nM T13201 C10GOE 397555 Ki = 3 nM T13201 C7HME8 439246 Ki > 10000 nM T13201 CA8C5N 439514 Ki = 5930 nM T13201 CC54LQ 450256 IC50 > 10000 nM T13201 C5IPL1 471796 Ki = 4265 nM T13201 C5HM8E 474578 Ki = 783 nM T13201 CL0M9Y 482317 Ki > 100000 nM T13201 CHF2Y9 493949 Ki = 384 nM T13201 C02DMG 504302 Ki = 56.1 nM T13201 CU7XE2 504303 Ki = 58.5 nM T13201 CNLT49 504304 Ki = 378 nM T13201 COGF52 516871 Ki = 200000 nM T13201 CC2V0U 517096 Ki = 700 nM T13201 CD8S2T 517441 Ki = 8400 nM T13201 C49CNT 519869 Ki = 680 nM T13201 C49LCW 519974 Ki > 100000 nM T13201 CU8MR5 520660 Ki = 8030 nM T13201 CQK9J0 522606 Ki > 200000000 nM T13201 C5OA7L 522689 Ki > 300000000 nM T13201 CJ7FR6 533728 Ki = 790 nM T13201 C24ASH 539731 Ki = 1838 nM T13201 C7EBA4 540544 Ki > 10000 nM T13201 CFU6X9 560256 Ki = 699 nM T13201 C3H5SW 562880 Ki = 105900 nM T13201 CPV28T 567846 Ki = 9.4 nM T13201 CGHE12 607195 Ki > 50000 nM T13201 CIK9S3 607305 Ki > 10000 nM T13201 CP3SF2 609637 Ki = 78 nM T13201 C5EA3O 638001 Ki = 2480 nM T13201 CNR94Z 640087 IC50 = 14290 nM T13201 C1DX6J 640625 Ki > 100000 nM T13201 CUMO27 643477 Ki = 68700 nM T13201 CH05FZ 648662 Ki > 10000 nM T13201 C6PTC3 658040 Ki > 50000 nM T13201 CS9F8K 667829 Ki = 47.2 nM T13201 CRTE89 667830 Ki = 34.1 nM T13201 CRZB53 669716 Ki = 13270 nM T13201 CU9ZY6 670087 Ki = 346 nM T13201 CYGK68 676946 Ki = 320 nM T13201 CMO61A 694792 Ki = 60 nM T13201 C4YWI2 702292 Ki = 29.6 nM T13201 CYZ9O5 703304 Ki > 10000 nM T13201 C9JH0M 706033 Ki > 50000 nM T13201 C7ZE6K 706849 Ki > 50000 nM T13201 CK7DO5 708535 Ki = 100 nM T13201 CK9HY0 716763 Ki > 1000 nM T13201 C8J4SO 724642 Ki = 81 nM T13201 C61NGE 724799 Ki = 586.5 nM T13201 CNTI96 728666 Ki = 63700 nM T13201 C8J7CO 730546 Ki = 35 nM T13201 C8G7EC 730672 Ki = 2150 nM T13201 COQ14K 738631 Ki = 52 nM T13201 CNJZ35 738819 Ki > 50000 nM T13201 CV6Y7U 740560 IC50 > 50000 nM T13201 CZM6W0 742873 Ki = 31.2 nM T13201 C3SAH9 743904 Ki = 40 nM T13201 CLG6H5 746816 Ki > 1000 nM T13201 CRIJ01 747569 Ki = 50 nM T13201 CW90GV 767467 Ki = 26.8 nM T13201 CV79DU 776418 Ki > 50000 nM T13201 CQJ06V 780268 IC50 = 197.64 nM T13201 CO1KN3 788171 Ki = 6.1 nM T13201 CA2B8X 792066 Ki > 50000 nM T13201 CM0VX3 809685 Ki = 922.5 nM T13201 CT0WB5 810867 Ki > 100000 nM T13201 C6LN8S 816982 Ki > 500000 nM T13201 C5BGW9 818267 Ki > 50000 nM T13201 CJP5D4 818647 IC50 > 50000 nM T13201 CVJZ57 818753 Ki > 50000 nM T13201 CF93TC 821388 Ki = 630 nM T13201 C5VJZ0 822776 Ki = 116 nM T13201 CTD64N 834412 Ki = 21.9 nM T13201 CHE97G 834460 IC50 = 120.13 nM T13201 CO31FL 853546 Ki = 56.7 nM T13201 C8SN5L 889524 Ki = 407 nM T13201 CQ45SF 892618 Ki = 125 nM T13201 CEN67I 897592 Ki = 4160 nM T13201 C51FVL 906840 Ki > 10000 nM T13201 CL2G3R 917163 Ki = 74 nM T13201 CKV7B6 917551 Ki = 2361 nM T13201 C4I3PJ 922062 Ki = 919.4 nM T13201 CRGQ70 927433 Ki = 47700 nM T13201 CO7XW0 928228 Ki > 10000 nM T13201 C6XQO2 940540 Ki > 50000 nM T13201 C4L9QD 943114 Ki > 10000 nM T13201 COH62A 943115 Ki > 10000 nM T13201 C7FI1J 970570 Ki = 135 nM T13201 CX3U0S 975396 Ki > 50000 nM T13201 CZ3WK7 983751 Ki = 28.3 nM T13201 CN71CV 989611 Ki > 10000 nM T13201 C4TE0N 990581 Ki = 12450 nM T13201 C5CED0 1014382 IC50 = 631.92 nM T13201 CXQ3M7 1016209 IC50 = 213.69 nM T13201 C6MU1W 1069008 Ki = 8350 nM T13201 CJ2S0M 1070919 Ki = 24.7 nM T13201 CYS9A2 1070922 Ki = 71 nM T13201 CM2C5N 1070928 Ki = 31.3 nM T13201 COM2R4 1070933 Ki = 47.1 nM T13201 CKA4R5 1080680 Ki = 8100 nM T13201 CDK1Z2 1085887 Ki > 50000 nM T13201 CA67JK 1124687 Ki > 1000 nM T13201 CZ04BL 1136487 IC50 = 126.47 nM T13201 C4QX1Z 1146666 Ki = 96.4 nM T13201 CWD7G1 1147802 Ki = 4230 nM T13201 CJ82NF 1178394 Ki = 465 nM T13201 C7A8VI 1211699 Ki = 26.1 nM T13201 CYF34N 1211700 Ki = 126 nM T13201 C7QP5E 1213792 Ki = 271 nM T13201 C6T0NU 1230924 Ki > 10000 nM T13201 C06ZSP 1234749 Ki = 15500 nM T13201 C9IBF8 1241259 Ki = 138 nM T13201 CF1N3S 1277269 Ki = 8550 nM T13201 CL87AM 1286568 Ki = 458 nM T13201 CA1I9S 1286583 Ki > 50000 nM T13201 CE6W7O 1287222 Ki > 10000 nM T13201 CP60YD 1294363 Ki = 210.7 nM T13201 CYGO97 1300832 IC50 = 660.65 nM T13201 C5XNB4 1307068 Ki > 10000 nM T13201 C40CKN 1316238 Ki = 2443 nM T13201 CDWO53 1346695 Ki = 9.7 nM T13201 CC3G1N 1377410 Ki > 50000 nM T13201 C9DY2L 1488548 Ki > 200000 nM T13201 CN5I0K 1505151 Ki > 50000 nM T13201 CAHP42 1548275 Ki = 324 nM T13201 C51SMF 1551768 Ki = 871 nM T13201 CORY25 1581900 Ki = 292.28 nM T13201 C4YUX5 1594254 Ki = 15000 nM T13201 C40YCV 1655994 Ki = 4002.6 nM T13201 CU7KR6 1738244 Ki > 10000 nM T13201 C7XSO5 1748172 Ki > 10000 nM T13201 CGKP07 1748225 Ki > 10000 nM T13201 C98OLG 1775694 Ki > 10000 nM T13201 C5PU0O 1809247 IC50 = 156.78 nM T13201 CJ4G3B 1817956 Ki = 260 nM T13201 C9ZEH2 1825978 IC50 = 16.73 nM T13201 CY20OQ 1945421 Ki = 678 nM T13201 CTF8R5 1957305 Ki > 100000 nM T13201 CR56WH 1968441 IC50 = 693.64 nM T13201 CK10DB 1977749 Ki = 187 nM T13201 C1DWG0 1989902 Ki = 67.1 nM T13201 CDQR23 2049187 Ki = 797 nM T13201 C45WTO 2059531 Ki = 24000 nM T13201 CSQJ97 2065546 Ki = 5142 nM T13201 CTK8C6 2089520 Ki > 50000 nM T13201 C93VNU 2089779 Ki = 324 nM T13201 C3W4PG 2192287 Ki = 37 nM T13201 C2O9YS 2196398 Ki = 220 nM T13201 C26OJZ 2206358 Ki = 50 nM T13201 CQS3A7 2207483 Ki > 10000 nM T13201 C3Y2CQ 2217668 Ki = 69 nM T13201 CO7JC2 2242987 Ki = 12 nM T13201 C3FIK2 2268367 Ki = 23000 nM T13201 CEW2Q3 2283723 Ki > 100000 nM T13201 COB96D 2305168 Ki = 86.4 nM T13201 C6FN0O 2316976 Ki = 446 nM T13201 CGW6L4 2318645 Ki > 100000 nM T13201 CD98QK 2333105 Ki = 834 nM T13201 C1V0KL 2357187 Ki = 52.4 nM T13201 C3BJ4K 2368995 Ki = 393 nM T13201 CTJ42W 2368997 Ki = 453 nM T13201 C4TD8M 2388085 Ki = 7.5 nM T13201 C1TW9F 2457081 Ki = 2479 nM T13201 CJ10IX 2470552 Ki = 31.5 nM T13201 CR65UH 2471990 Ki > 50000 nM T13201 C95INQ 2476733 Ki = 10.9 nM T13201 C75SLD 2496330 Ki = 3.7 nM T13201 C2H4KT 2520594 Ki = 41.3 nM T13201 CBN52G 2566555 Ki = 24 nM T13201 CO1PU5 2570886 Ki = 21 nM T13201 CKH53Q 2723810 Ki = 1040000 nM T13201 C8YH7W 2733779 Ki = 1000 nM T13201 C0V7XB 2733782 Ki > 100000 nM T13201 C0W8UL 2735045 Ki = 604 nM T13201 CQ70UR 2755708 Ki = 17.9 nM T13201 CU60ZB 2755709 Ki = 20 nM T13201 CNG69U 2755712 Ki = 21.5 nM T13201 C58ISM 2755728 Ki = 48.7 nM T13201 C8QGL9 2760606 Ki > 10000 nM T13201 CNGK51 2781602 Ki = 5800 nM T13201 CS0R6B 2789347 Ki > 10000 nM T13201 CD41AE 2795990 Ki = 6250 nM T13201 CCOI52 2797418 Ki = 129 nM T13201 C21FUI 2801263 Ki = 14480 nM T13201 C4IDC5 2809317 Ki = 410000 nM T13201 C4V0MQ 2812911 Ki = 10750 nM T13201 CPO6W3 2813478 Ki = 9.7 nM T13201 CUI4Y8 2814914 Ki = 1106 nM T13201 CLFB40 2815883 Ki > 10000 nM T13201 CDSN81 2826269 Ki = 72.3 nM T13201 CEY4J6 2858793 IC50 = 36.13 nM T13201 CU6D3W 2881615 IC50 > 10000 nM T13201 CBPO81 2882281 Ki = 266 nM T13201 CVA6F2 2893744 IC50 > 10000 nM T13201 CE2GR3 2900806 Ki > 500000 nM T13201 CME74N 2904589 Ki = 1710 nM T13201 CW9M7A 2952488 Ki > 50000 nM T13201 CFO90D 2952737 Ki > 50000 nM T13201 CQ9T8W 2970501 Ki = 66 nM T13201 C61OTP 2991092 Ki = 437 nM T13201 CFV92S 3000601 Ki = 610 nM T13201 CZEH20 3003616 Ki = 47.4 nM T13201 CJ9LZ7 3051101 Ki = 72000 nM T13201 CN2Y5M 3083616 Ki = 9890 nM T13201 C9GT5Z 3083928 Ki = 9.7 nM T13201 CY0OZ3 3090044 Ki = 79 nM T13201 C84TYH 3108089 IC50 = 231.41 nM T13201 CY19CS 3115791 Ki = 96.9 nM T13201 C49VDN 3132886 Ki = 412 nM T13201 CQI7A2 3133127 Ki = 318 nM T13201 CP58HK 3344056 Ki = 980 nM T13201 C6V3ES 3365615 Ki = 55 nM T13201 CXU4J8 3377675 Ki = 102 nM T13201 C1K6IA 3379075 Ki = 109 nM T13201 C0FV7M 3414913 Ki = 1000 nM T13201 CL6E2Y 3426384 Ki = 6445 nM T13201 CT1NB8 3441996 Ki = 9 nM T13201 CZW71J 3476048 IC50 = 503.74 nM T13201 CP3BS4 3489403 Ki = 40 nM T13201 CHM17U 3496881 Ki = 8510 nM T13201 CIXH89 3516083 Ki = 8.6 nM T13201 C0VI6O 3524248 Ki > 50000 nM T13201 CM6R3S 3525535 Ki = 30 nM T13201 CKTY04 3538605 Ki = 0.96 nM T13201 C86GSL 3542746 Ki = 380 nM T13201 CHGS79 3551941 Ki = 3713.2 nM T13201 CDI8T5 3576817 Ki = 7700 nM T13201 C9L1HS 3586494 Ki = 28.5 nM T13201 CS5Z1Q 3614018 Ki = 1290 nM T13201 CD0FL4 3627258 Ki = 87 nM T13201 CS4TM2 3638938 Ki = 2000 nM T13201 CY89AI 3649509 Ki = 8600 nM T13201 C4WZG2 3657160 Ki > 50000 nM T13201 CDY79J 3669864 Ki = 55300 nM T13201 CBED02 3683067 Ki = 13000 nM T13201 C3REH6 3703019 IC50 > 50000 nM T13201 CQ5F9P 3724005 Ki = 246 nM T13201 CF9VG2 3770187 Ki = 9435 nM T13201 CLW43B 3813634 Ki = 6352 nM T13201 C2SY4L 3856570 Ki > 10000 nM T13201 CI3KT8 3936209 Ki > 10000 nM T13201 CV0KG3 3950536 Ki > 10000 nM T13201 CJ6D2S 3970972 Ki = 109 nM T13201 C8C4DV 4053995 Ki = 6300 nM T13201 C5T1YZ 4056562 Ki = 8100 nM T13201 C37VWB 4070422 Ki = 12500 nM T13201 C25EPG 4073057 Ki = 32 nM T13201 C3CGU6 4094683 Ki = 72 nM T13201 CU2O1Y 4110011 Ki = 165500 nM T13201 C8DZ4B 4121769 Ki = 9.4 nM T13201 C9O0GV 4158561 Ki = 153 nM T13201 CPA56O 4180608 Ki = 950 nM T13201 CDNL69 4184455 Ki = 137800 nM T13201 CT57HM 4204917 Ki > 10000 nM T13201 CHOE81 4218706 Ki = 47 nM T13201 CORC17 4228388 Ki = 50 nM T13201 CD2P7T 4259683 Ki = 210 nM T13201 CV6BJ7 4262171 Ki = 33550 nM T13201 CUT26E 4274816 Ki > 50000 nM T13201 CUE97L 4276695 Ki > 10000 nM T13201 C5PM3E 4321567 Ki = 640000 nM T13201 CQ3P4I 4323207 Ki = 7 nM T13201 CI7UR5 4343483 Ki > 200000000 nM T13201 CI6AE7 4377996 Ki = 7000 nM T13201 CQ2X7N 4389798 Ki = 24 nM T13201 C4E5VQ 4447263 Ki = 339 nM T13201 C96LCZ 4476238 Ki = 2280 nM T13201 CIF43A 4572067 Ki = 69 nM T13201 CJ63TI 4578038 Ki = 4.9 nM T13201 CE5LO8 4578265 Ki = 2587.3 nM T13201 C7RS2F 4583704 Ki > 1000 nM T13201 CAPM27 4598704 Ki > 50000 nM T13201 C3Q1WN 4607842 Ki = 92 nM T13201 CDK4L0 4608376 Ki = 540000 nM T13201 C02JOA 4616277 Ki = 81300 nM T13201 CCP96V 4617978 Ki = 1000 nM T13201 C6XVK9 4619076 Ki = 7450 nM T13201 CLSY09 4626049 Ki = 670 nM T13201 CLQ7U4 4627354 IC50 = 423.42 nM T13201 C3GDR0 4634582 Ki = 2100 nM T13201 CW1A4Z 4637857 Ki = 59 nM T13201 CPX3W6 4650747 Ki = 364 nM T13201 CTM71V 4654716 Ki = 341 nM T13201 CCB9Z5 4656684 Ki = 82 nM T13201 C2WI3U 4667972 Ki = 124 nM T13201 C07MRI 4712722 Ki = 200000 nM T13201 CWXE71 4718084 Ki = 4.3 nM T13201 C6RC3L 4718087 Ki = 4.5 nM T13201 C5FZ0L 4718107 IC50 = 172.84 nM T13201 CRL7B4 4718142 Ki = 15.5 nM T13201 CJM5F3 4718971 Ki = 4.6 nM T13201 CAG10X 4723337 IC50 = 258.84 nM T13201 C6B0OY 4723880 Ki = 15.6 nM T13201 C0MFT8 4801151 Ki = 1368 nM T13201 CSC7B8 4803242 Ki = 275 nM T13201 CUA65R 4857564 Ki = 494 nM T13201 CX8C3P 4961927 Ki = 78.5 nM T13201 CX3RJ9 5005133 Ki = 351 nM T13201 CIP6Q8 5017140 Ki = 41.5 nM T13201 C7JBU0 5019114 Ki = 527 nM T13201 CF94ER 5032527 Ki > 10000 nM T13201 CD9V5J 5044227 Ki = 4810 nM T13201 C49FDN 5046067 Ki = 143 nM T13201 CTB04Y 5050031 Ki = 10000 nM T13201 CX60DM 5067385 Ki = 1390 nM T13201 C4OAL9 5070078 Ki = 6300 nM T13201 CN31CX 5071527 Ki = 386 nM T13201 CSG29M 5073140 Ki = 55 nM T13201 CU8E4B 5133468 Ki = 43200 nM T13201 C7GXU1 5147921 Ki = 11000000 nM T13201 C89OCE 5155717 Ki = 212 nM T13201 CM9N8G 5161767 Ki > 10000 nM T13201 C6HM0R 5164092 Ki = 7520 nM T13201 C4HB1G 5172319 Ki = 50 nM T13201 CI8JY0 5172475 Ki = 9300 nM T13201 CC37SW 5182516 Ki = 12500 nM T13201 CZBY34 5220706 Ki = 15000 nM T13201 CY9IV8 5223338 Ki = 9.7 nM T13201 CEN0L7 5227639 Ki = 63 nM T13201 CFQ62G 5232078 Ki > 100000 nM T13201 CEBD92 5272990 Ki = 63600 nM T13201 CP09FG 5272997 Ki = 29600 nM T13201 C4SV5T 5273568 Ki = 5040 nM T13201 CU4E5S 5273569 Ki = 4860 nM T13201 CZS0G5 5276565 IC50 = 7136 nM T13201 C3JN0F 5277465 IC50 > 10000 nM T13201 CRJK67 5277481 IC50 = 8285 nM T13201 CYF7S5 5277490 IC50 = 814 nM T13201 CD1LZ7 5278580 Ki = 26.9 nM T13201 CNZ73E 5280567 Ki > 100000 nM T13201 CN10FM 5281793 Ki > 10000 nM T13201 CA18OQ 5316302 Ki = 36400 nM T13201 CTJ01E 5317485 Ki = 5600 nM T13201 CI58XK 5319562 Ki = 780 nM T13201 CNO53D 5321265 Ki = 7660 nM T13201 CP0R5H 5336569 Ki > 10000 nM T13201 C8PS4E 5358858 Ki = 7810 nM T13201 C4KHR2 5431473 IC50 = 3.09 nM T13201 CRVS37 5449904 Ki > 10000 nM T13201 C2UN6J 5462815 Ki = 540000 nM T13201 CH5OM1 5463917 Ki = 22500000 nM T13201 CG76KE 5470394 Ki = 1 nM T13201 CXEW32 5491996 Ki = 6450 nM T13201 C7RG3L 5496307 Ki = 3350 nM T13201 CX71JE 5682293 Ki > 10000 nM T13201 CWYU91 5742696 Ki = 5070 nM T13201 CU0FW5 5743063 Ki = 2780 nM T13201 C4VZP8 5765787 Ki = 40 nM T13201 CWL5R2 5765789 Ki = 32.9 nM T13201 CK0M4A 5910585 Ki = 9750 nM T13201 C7T1DV 5956379 Ki = 1 nM T13201 CHJ3V8 6102658 Ki > 100000 nM T13201 CJZ47Y 6365232 Ki = 8500 nM T13201 CS4KQ6 6482974 Ki = 4310 nM T13201 C9L8AX 6537802 Ki = 9 nM T13201 C65FRB 6852128 Ki = 7 nM T13201 CPFV65 6916013 Ki = 33 nM T13201 CK85ZF 7022526 IC50 > 50000 nM T13201 C0W5GD 7130726 Ki = 482.1 nM T13201 CWL9C2 7382212 Ki > 10000 nM T13201 C75SBG 7382231 Ki > 50000 nM T13201 C6U9MT 7382238 Ki > 50000 nM T13201 CY57CX 7382249 Ki = 3579 nM T13201 C5TK0N 7463363 IC50 = 4870 nM T13201 C7RM6F 7463364 IC50 = 7660 nM T13201 C9UJB7 7463369 IC50 = 8060 nM T13201 CKCM96 7463376 Ki = 1250 nM T13201 CDCP43 7766335 Ki > 50000 nM T13201 CTH8D3 7785988 Ki = 43.9 nM T13201 C95AKP 7794397 Ki = 1503 nM T13201 C6S5HK 7832430 Ki = 208 nM T13201 C1EKW8 7996519 Ki > 40000 nM T13201 C6WG0N 8007128 Ki = 24 nM T13201 C67SFK 8084575 Ki > 50000 nM T13201 CQ0Z4E 8098235 Ki = 240 nM T13201 CCW8R6 8190912 Ki = 9620 nM T13201 CSW01Z 8272034 Ki = 1480 nM T13201 C9BAM4 8281641 Ki = 38.8 nM T13201 C3WQ9M 8866559 Ki = 42.4 nM T13201 C5CS1Y 9314410 Ki = 314.2 nM T13201 C3SA2N 9314413 Ki = 374.4 nM T13201 C47VSJ 9572721 Ki = 379000 nM T13201 CIJ25V 9794947 IC50 = 7680 nM T13201 C7SRM4 9837496 IC50 = 7890 nM T13201 C0EJ1Q 9847197 Ki = 10 nM T13201 C6YW0Q 9942868 Ki = 116.4 nM T13201 CSIY73 9952009 IC50 > 100000 nM T13201 CJS4I3 9990000 Ki = 760 nM T13201 CIN68V 9998184 Ki = 110 nM T13201 CY47OI 9998322 Ki = 95 nM T13201 C6TO0A 10001582 Ki = 90 nM T13201 CXD28H 10015065 Ki = 7.3 nM T13201 CNKD31 10016330 Ki = 2324 nM T13201 C4UEV9 10016475 Ki > 10000 nM T13201 CF6RN0 10018880 Ki = 120 nM T13201 CX4MK5 10019750 Ki = 9000 nM T13201 CKOV96 10023066 Ki = 29 nM T13201 CQL10G 10026448 Ki = 12 nM T13201 C6DGR7 10027203 Ki > 200 nM T13201 CX2W9O 10037048 IC50 = 6780 nM T13201 CO39PK 10042482 Ki = 7 nM T13201 CI5AR1 10044828 Ki = 36 nM T13201 C5Q1FI 10052644 Ki = 5 nM T13201 C5X7GY 10059582 Ki = 2541 nM T13201 CWM01R 10059806 Ki = 18356 nM T13201 COWD07 10062976 Ki = 170 nM T13201 C69DPZ 10068042 IC50 > 10000 nM T13201 C6FKM3 10069411 Ki = 13 nM T13201 CY8F0E 10076040 Ki = 40100 nM T13201 CU7DJ1 10081163 Ki = 51000 nM T13201 C0P5XV 10081897 Ki = 1066 nM T13201 CD58EL 10083644 Ki > 50000 nM T13201 CCR24T 10087045 Ki = 350 nM T13201 CZU5A2 10088969 Ki = 27 nM T13201 CRN29P 10104483 Ki = 4.6 nM T13201 C7WU0A 10107532 Ki = 4403 nM T13201 CAQ6I1 10131078 Ki = 63 nM T13201 CXD91O 10136406 Ki = 19.1 nM T13201 CVRZ27 10198038 IC50 = 8790 nM T13201 C63AZQ 10198750 Ki = 75 nM T13201 CUR4O7 10198795 Ki = 72 nM T13201 CJV68L 10220266 Ki = 930.2 nM T13201 CM4E8G 10243877 Ki = 6 nM T13201 C4E1JQ 10245883 Ki = 185 nM T13201 CX50AK 10266719 Ki = 22500 nM T13201 CC9XT4 10267015 Ki = 630 nM T13201 CLM6Z5 10290835 Ki = 690000 nM T13201 CS3CE7 10313432 Ki = 15 nM T13201 CQ8A0I 10328097 Ki > 10000 nM T13201 CN40WD 10331524 Ki = 1864 nM T13201 CU9OI5 10334780 Ki = 6 nM T13201 CUE81P 10337354 Ki = 1347 nM T13201 CRHU49 10338639 Ki = 360 nM T13201 CX6P1I 10358994 Ki = 3 nM T13201 CH4I9P 10360342 Ki = 620 nM T13201 C58IYR 10366827 Ki = 1670 nM T13201 C3HBY6 10375558 Ki = 185 nM T13201 CT9VJ3 10383097 Ki = 975 nM T13201 C1O2FH 10383098 Ki = 1700 nM T13201 CP2XW6 10387325 Ki = 2000 nM T13201 CVW18K 10409391 Ki = 5 nM T13201 C5IK7H 10420920 Ki = 40 nM T13201 C4MI8O 10423003 Ki = 270 nM T13201 CI60TB 10423771 Ki = 6 nM T13201 CFGK83 10430595 Ki = 13 nM T13201 CVIN94 10439991 Ki > 10000 nM T13201 CIC54M 10452478 Ki = 420 nM T13201 C6T8VC 10456675 Ki = 150 nM T13201 CED61Q 10467688 Ki = 500 nM T13201 C6TYP0 10467861 Ki > 10000 nM T13201 C25NJB 10471772 Ki = 4007 nM T13201 C13JVK 10477954 Ki = 2000 nM T13201 CEV92X 10493372 Ki = 14600 nM T13201 C41KHC 10494655 Ki = 47 nM T13201 CJFC96 10495006 Ki = 21 nM T13201 C4ZV9X 10495711 Ki = 45 nM T13201 C3Y0AX 10497272 Ki = 510 nM T13201 CE2XQ6 10497552 Ki = 16 nM T13201 CPMT67 10497717 Ki = 21 nM T13201 CSZ1K0 10499069 Ki = 21 nM T13201 CL8O6I 10500340 Ki = 21 nM T13201 CVID65 10500886 Ki > 200 nM T13201 CBL23S 10502993 Ki = 370 nM T13201 CV0FT4 10503780 Ki = 750 nM T13201 CA95ZO 10504238 Ki = 805 nM T13201 CU8E4S 10505384 Ki = 5000 nM T13201 CRS2V1 10505991 Ki = 43000 nM T13201 CRJ8O1 10506509 Ki = 12 nM T13201 CH6A2O 10507009 Ki = 112000 nM T13201 C3TCR7 10507836 Ki = 615 nM T13201 CRNO69 10508249 Ki = 41 nM T13201 CR3AL4 10508270 Ki = 1850 nM T13201 CG0MZ8 10508351 Ki = 330 nM T13201 C52EMX 10509011 Ki = 4400 nM T13201 CIW1L8 10509163 Ki = 300 nM T13201 C3G4PQ 10509380 Ki = 7000 nM T13201 CD41CA 10512636 Ki = 851.7 nM T13201 CJZ67W 10515762 Ki = 110 nM T13201 CR63LA 10518811 Ki = 190 nM T13201 CFOE60 10519650 Ki = 155500 nM T13201 CM0K8P 10519868 Ki = 21 nM T13201 CXD8I5 10523292 Ki = 18 nM T13201 CZT6S0 10523695 Ki = 53 nM T13201 CU2E3A 10524550 Ki = 14 nM T13201 CZ4LU8 10524990 Ki = 360 nM T13201 CQL8S4 10525380 Ki = 12 nM T13201 C7UY4Z 10526065 Ki = 47 nM T13201 CM4Q7C 10526660 Ki = 300 nM T13201 CUJI62 10527611 Ki = 5500 nM T13201 C7Z1LE 10527692 Ki = 22000 nM T13201 CK43UF 10528302 Ki = 24500 nM T13201 CG1M8V 10529267 Ki = 25300 nM T13201 CGK37L 10529602 Ki > 200 nM T13201 CI6SU7 10530110 Ki = 1100 nM T13201 CTP62O 10530164 Ki = 52 nM T13201 CU6HX8 10530223 Ki = 18000 nM T13201 C6C7YQ 10531119 Ki = 290000 nM T13201 CA5C0S 10531121 Ki = 92000 nM T13201 CND17Q 10532205 Ki = 300 nM T13201 C3PO6V 10532224 Ki = 47 nM T13201 CC0EB5 10532491 Ki = 400 nM T13201 CU6YM4 10532987 Ki = 2550 nM T13201 CJ1D2U 10533054 Ki = 3000 nM T13201 CWQY26 10535227 Ki > 10000 nM T13201 CT04WN 10537366 Ki = 25000 nM T13201 C5PMH4 10539133 Ki = 22000 nM T13201 C5G8EX 10540518 Ki = 510 nM T13201 C5I3JC 10541189 Ki = 15000 nM T13201 C9EM7W 10543041 Ki = 39 nM T13201 C3KHS0 10543744 Ki = 540 nM T13201 C81ZYH 10543818 Ki = 61 nM T13201 C5S9PM 10546426 Ki = 12 nM T13201 CIN60X 10548978 Ki = 19 nM T13201 C0S7OI 10549020 Ki = 1080 nM T13201 C5JS8L 10549329 Ki > 200 nM T13201 CY93AQ 10549606 Ki = 590 nM T13201 CN8KT4 10550727 Ki = 525 nM T13201 C3ALP8 10550907 Ki = 1450 nM T13201 CCTN57 10551138 Ki = 54 nM T13201 CQ2U6H 10552761 Ki = 200 nM T13201 C31INC 10553159 Ki = 2560 nM T13201 C8CJ3W 10554523 Ki = 40000 nM T13201 C9CHQ8 10554752 Ki = 1500 nM T13201 C4C5YD 10555371 Ki = 35 nM T13201 CDJ9O6 10555708 Ki = 12 nM T13201 C6QH5Y 10555828 Ki = 1400 nM T13201 CJ74IY 10556211 Ki = 620 nM T13201 CVJ85T 10556224 Ki = 41 nM T13201 CV79UJ 10556471 Ki = 43 nM T13201 C08EWG 10563541 Ki = 600 nM T13201 CQP6G1 10565056 Ki = 20300 nM T13201 CCKE29 10566405 Ki = 175000 nM T13201 C7UYX1 10566734 Ki = 280 nM T13201 C7U2DR 10567673 Ki = 510 nM T13201 CLFN25 10567759 Ki = 15000 nM T13201 C3W9QA 10568362 Ki = 110 nM T13201 CD8T0J 10568499 Ki = 23 nM T13201 CT6BA5 10572515 Ki = 5000 nM T13201 C8RD4P 10573046 Ki = 575 nM T13201 CP71JY 10573928 Ki = 790 nM T13201 CRO7J0 10574278 Ki = 120 nM T13201 C2PH8Q 10575017 Ki = 90 nM T13201 C9N8YQ 10575994 Ki = 360 nM T13201 CQ3XL8 10576231 Ki = 65 nM T13201 C8CMG3 10577063 Ki = 13 nM T13201 CF3A4I 10577600 Ki = 12000 nM T13201 CN8R3Y 10577727 Ki = 1900 nM T13201 CQV65S 10578334 Ki = 1700 nM T13201 C6CNQ7 10578619 Ki = 750 nM T13201 CCNW04 10578621 Ki = 30500 nM T13201 C6HO9B 10578774 Ki = 300 nM T13201 C8I9FB 10580194 Ki = 10 nM T13201 C28OGL 10580382 Ki = 37 nM T13201 C8UW9L 10580477 Ki = 2480 nM T13201 C9CF5Q 10580554 Ki = 300 nM T13201 CJ8IW3 10581021 Ki = 890 nM T13201 CAVB38 10586310 Ki = 16600 nM T13201 C73KXU 10586607 Ki = 213000 nM T13201 C0BPD3 10589291 Ki = 17 nM T13201 CD4V5G 10590334 Ki = 10 nM T13201 C0N1IM 10590553 Ki = 54 nM T13201 C6KD1Z 10591288 Ki = 775 nM T13201 C8J6HS 10591505 Ki = 50 nM T13201 CB20LM 10594000 Ki > 200 nM T13201 C25DOL 10594934 Ki = 21 nM T13201 CBM48L 10596042 Ki = 605 nM T13201 CAZ36G 10596413 Ki = 270 nM T13201 C1JRL7 10597208 Ki = 890 nM T13201 CH37KM 10599305 Ki = 300 nM T13201 C3VZX6 10599546 Ki = 1500 nM T13201 CAL87S 10599609 Ki = 1800 nM T13201 CH6J5O 10600355 Ki = 680 nM T13201 CY8HT7 10601085 Ki = 10200 nM T13201 C8LE1Z 10601296 Ki = 325 nM T13201 CO8D2C 10602116 Ki = 6000 nM T13201 CM6I8S 10602258 Ki = 1500 nM T13201 CWG1C7 10602601 Ki = 1600 nM T13201 CZB76C 10602667 Ki = 6000 nM T13201 CP4AY9 10603234 Ki = 600 nM T13201 C9SLH3 10603241 Ki = 33 nM T13201 C9YR2K 10603335 Ki = 320 nM T13201 CJNP46 10603338 Ki = 1650 nM T13201 C6G0ZI 10603469 Ki = 61 nM T13201 C6C9ZB 10603761 Ki = 4000 nM T13201 CT4EC1 10603881 Ki = 1600 nM T13201 C73UOS 10604129 Ki = 350 nM T13201 C65GKZ 10609913 Ki = 350 nM T13201 C5G9MI 10610114 Ki = 33000 nM T13201 CZS6O0 10610757 Ki = 305 nM T13201 CN38WB 10611730 Ki = 290 nM T13201 C8N4EO 10614528 Ki = 800 nM T13201 C2PRM1 10615166 Ki = 800 nM T13201 CM46AO 10615795 Ki = 100000 nM T13201 C78TRD 10617314 Ki = 360 nM T13201 C1EIP0 10618881 Ki = 1560 nM T13201 CF85VP 10620016 Ki = 760 nM T13201 CSY79P 10620807 Ki = 8000 nM T13201 CM9H5A 10623288 Ki = 600 nM T13201 C8HRI3 10623948 Ki = 1700 nM T13201 C97JCY 10625036 Ki = 10000 nM T13201 CU3YT8 10625038 Ki = 1000 nM T13201 CVN72J 10625060 Ki = 13000 nM T13201 C4FLA9 10625484 Ki = 24000 nM T13201 CGI03J 10625651 Ki = 265000 nM T13201 CMQC23 10625732 Ki = 200 nM T13201 CGB5S0 10626619 Ki = 94000 nM T13201 CCX2K6 10627219 Ki = 55 nM T13201 CWN3O4 10628503 Ki = 470 nM T13201 C9N2ZH 10629041 Ki = 3400 nM T13201 CFL47V 10629052 Ki = 600 nM T13201 C9TSQ6 10632698 Ki = 9200 nM T13201 C4I2QF 10633163 Ki = 15000 nM T13201 C2OHP3 10635833 Ki = 820 nM T13201 C0KA3F 10637879 Ki = 950 nM T13201 C7YOD1 10637941 Ki = 20800 nM T13201 C4VQC3 10638194 Ki = 188400 nM T13201 CU6IE1 10640069 Ki = 36 nM T13201 CPH72T 10640797 Ki = 180000 nM T13201 CN6HA4 10642039 Ki = 350 nM T13201 CJV5L1 10643532 Ki = 1500 nM T13201 CC8T9S 10645605 Ki = 600 nM T13201 CNAE38 10647590 Ki = 41 nM T13201 CIW58E 10648512 Ki = 20900 nM T13201 C9V3WZ 10649387 Ki = 54 nM T13201 CCI16T 10649726 Ki = 15000 nM T13201 CK2F6I 10649728 Ki = 27500 nM T13201 CQB3T1 10650115 Ki = 4 nM T13201 CG4HL1 10650150 Ki = 750 nM T13201 CZN6S5 10650429 Ki = 19 nM T13201 CC4UM6 10650450 Ki = 110000 nM T13201 CW2AC6 10651479 Ki = 900 nM T13201 CZ9GS7 10651537 Ki = 610 nM T13201 CSV84J 10651858 Ki = 38 nM T13201 CFJA05 10651893 Ki = 1400 nM T13201 CE14NG 10652046 Ki = 15000 nM T13201 CE24FZ 10660854 Ki = 17000 nM T13201 CIMZ90 10663338 Ki = 21500 nM T13201 C19DBM 10663960 Ki = 44 nM T13201 C4SX7R 10665257 Ki = 54 nM T13201 C6VBM9 10665468 Ki = 550 nM T13201 CMN37R 10666283 Ki = 70 nM T13201 CC8WH4 10666501 Ki = 570 nM T13201 C3E0ZP 10667414 Ki = 60 nM T13201 C9IL3M 10670278 Ki = 760 nM T13201 C1W7CO 10671070 Ki = 11000 nM T13201 CB39ZS 10671185 Ki = 35000 nM T13201 CWB19K 10671441 Ki = 127 nM T13201 CWQ58H 10671476 Ki = 330 nM T13201 CB6CA9 10672102 Ki = 1070 nM T13201 CQK8V3 10673297 Ki = 26000 nM T13201 CVX50Z 10673405 Ki = 300 nM T13201 CJ9D7F 10673563 Ki = 8000 nM T13201 C6AH3Z 10673625 Ki = 720 nM T13201 CETF96 10673746 Ki = 125000 nM T13201 C79OXJ 10673953 Ki = 1400 nM T13201 CY9W0O 10674571 Ki = 750 nM T13201 C02FIM 10674633 Ki = 300 nM T13201 CL6GZ4 10675046 Ki = 9 nM T13201 CR2D8E 10675795 Ki = 1500 nM T13201 C6B8JA 10675931 Ki = 1000 nM T13201 CSZ39G 10676062 Ki = 22000 nM T13201 CS2FT7 10676818 Ki = 8000 nM T13201 C9IAB0 10685830 Ki = 21000 nM T13201 C2UH7Z 10687216 Ki = 18500 nM T13201 CGJ7L6 10691042 Ki = 18 nM T13201 CVHO36 10692638 Ki = 900 nM T13201 C4BQK5 10693598 Ki = 105 nM T13201 C17ICZ 10693904 Ki = 210000 nM T13201 C0TOK2 10695275 Ki = 25 nM T13201 CHG04R 10695589 Ki = 13000 nM T13201 CH63NB 10695632 Ki = 15000 nM T13201 C2YH7O 10696741 Ki = 40000 nM T13201 CRL2U7 10696743 Ki = 280000 nM T13201 CE82AF 10697359 Ki = 7000 nM T13201 CV2RJ5 10697379 Ki = 21800 nM T13201 C0VF5D 10697562 Ki = 20300 nM T13201 CT59ZG 10697685 Ki = 28000 nM T13201 C0NM4D 10698231 Ki = 1770 nM T13201 C6MG9R 10698477 Ki = 11 nM T13201 C1P2SH 10698664 Ki = 270000 nM T13201 CKV21F 10699169 Ki = 10 nM T13201 C62VLP 10699783 Ki = 12 nM T13201 CXZ97V 10699991 Ki = 49 nM T13201 C0DIN6 10700505 Ki = 900 nM T13201 C5WSA3 10704587 Ki = 18000 nM T13201 C5E8QF 10707457 Ki = 32 nM T13201 CFZ65M 10710739 Ki = 135000 nM T13201 C8NH6B 10711889 Ki = 20600 nM T13201 C6D2TJ 10712038 Ki = 3450 nM T13201 CE8L3N 10712383 Ki = 35 nM T13201 C9LD0S 10712555 Ki = 22 nM T13201 CLV42Z 10713226 Ki = 600 nM T13201 C9PXS4 10714881 Ki = 98 nM T13201 CGNP20 10715470 Ki = 520 nM T13201 C23LAY 10715903 Ki = 310 nM T13201 C7JS2I 10716079 Ki = 1100 nM T13201 CX8YI4 10716240 Ki = 3000 nM T13201 CI6Y4G 10716883 Ki = 550 nM T13201 C3TGW8 10717400 Ki = 36 nM T13201 CG3NP5 10718314 Ki = 12 nM T13201 CDV6R8 10718340 Ki = 13 nM T13201 CS9X0E 10719552 Ki = 1000 nM T13201 CSJ14E 10720061 Ki = 19600 nM T13201 C1L8UA 10720537 Ki = 29 nM T13201 C8WJK7 10721281 Ki = 300 nM T13201 CB59QH 10721415 Ki = 23100 nM T13201 CT87NP 10721547 Ki = 150 nM T13201 CNF6H0 10721639 Ki = 290000 nM T13201 CT65DL 10722417 Ki = 13 nM T13201 C2OYQ1 10722508 Ki = 45 nM T13201 C3K1DN 10722521 Ki = 1800 nM T13201 C4VOP2 10722619 Ki = 300 nM T13201 C42TPS 10722680 Ki = 645 nM T13201 CSE58B 10723137 Ki = 310 nM T13201 CV9A8J 10723227 Ki = 965 nM T13201 C4GX0Y 10723329 Ki = 59 nM T13201 CR0M8G 10723505 Ki = 28 nM T13201 C2A6LI 10728925 Ki = 20300 nM T13201 CR5U3C 10734581 Ki = 540 nM T13201 CGX10J 10736890 Ki = 610 nM T13201 C2ZLE4 10737428 Ki = 198 nM T13201 C5G2OP 10737443 Ki = 27 nM T13201 C83KNR 10737789 Ki = 560 nM T13201 CL5U3V 10738713 Ki = 200000 nM T13201 CGH3P0 10738795 Ki = 62 nM T13201 CGTX61 10738796 Ki = 60 nM T13201 C8Z9IL 10739376 Ki = 900 nM T13201 CNW7S5 10740344 Ki = 545 nM T13201 C4FWC9 10740485 Ki = 29 nM T13201 CB9T4M 10742338 Ki = 15200 nM T13201 CN30YJ 10742576 Ki = 4000 nM T13201 CBF1Z5 10742874 Ki = 1000 nM T13201 CEBQ21 10744110 Ki = 18 nM T13201 CCRG49 10744718 Ki = 1755 nM T13201 C6O7PQ 10744771 Ki = 600 nM T13201 CW6Q1M 10744854 Ki = 300 nM T13201 C7WHI1 10745371 Ki = 300000 nM T13201 CG4OI8 10745793 Ki = 775 nM T13201 C0KN7Z 10745795 Ki = 23400 nM T13201 C6IP0J 10746098 Ki = 15 nM T13201 CTG8L5 10746646 Ki = 1400 nM T13201 CLMA04 10747000 Ki = 1680 nM T13201 CG8K9X 10747080 Ki = 630 nM T13201 CG1MT4 10747258 Ki = 2500 nM T13201 C0OC6N 10747270 Ki = 310 nM T13201 CXE89A 10747447 Ki = 24 nM T13201 C7BSK4 10747629 Ki = 4500 nM T13201 C8DL1Z 10747766 Ki = 2400 nM T13201 CY1WX7 10747964 Ki = 3000 nM T13201 CB6M3O 10747965 Ki = 3600 nM T13201 C7MEP5 10752797 Ki = 25500 nM T13201 CRG5Z7 10753241 Ki = 335 nM T13201 CB7T3Q 10755646 Ki = 49.4 nM T13201 CO8B6L 10756624 Ki = 1360 nM T13201 CA3F1N 10758013 Ki = 7 nM T13201 CQUP90 10759040 Ki = 80000 nM T13201 C14QMV 10759047 Ki = 1100 nM T13201 CY4RA2 10759222 Ki = 860 nM T13201 CA5BQ1 10763396 Ki = 50 nM T13201 CBHI21 10763843 Ki = 50 nM T13201 C3HVQ9 10764510 Ki = 6000 nM T13201 CTK7W3 10765251 Ki = 16000 nM T13201 CZ8S0A 10765253 Ki = 24000 nM T13201 CR4J2Z 10765565 Ki = 46 nM T13201 C4R2FB 10765728 Ki = 1870 nM T13201 C0XNP9 10765735 Ki = 300 nM T13201 CXD7E4 10765823 Ki = 7 nM T13201 CH78WD 10766083 Ki = 4000 nM T13201 CF5I7H 10766126 Ki = 18400 nM T13201 C69MAB 10766339 Ki = 5000 nM T13201 CA6C0Z 10766622 Ki = 100 nM T13201 CIB3E5 10766650 Ki = 6000 nM T13201 C06MYS 10766652 Ki = 1000 nM T13201 CVD0H3 10766865 Ki = 400 nM T13201 C96BYJ 10767057 Ki = 750 nM T13201 C2K3XN 10767400 Ki = 15 nM T13201 CM8JR1 10767828 Ki = 205 nM T13201 C9Z3EL 10767989 Ki = 1250 nM T13201 CRS6F0 10768100 Ki = 43 nM T13201 C7X3PW 10768529 Ki = 140000 nM T13201 C3L4OV 10768593 Ki = 300 nM T13201 CHVB87 10768870 Ki = 112000 nM T13201 CMS9R1 10769153 Ki = 125 nM T13201 C4CT1D 10769199 Ki = 810 nM T13201 CQ15VI 10769549 Ki = 21 nM T13201 CZDJ14 10770028 Ki = 350 nM T13201 C06DZW 10770030 Ki = 3600 nM T13201 CD4VK5 10770656 Ki = 400 nM T13201 CDU8X0 10770816 Ki = 46 nM T13201 CYG79W 10779489 Ki = 16200 nM T13201 C1T9VB 10782719 Ki = 845 nM T13201 C40YHF 10783082 Ki = 60 nM T13201 CRXH95 10784749 Ki = 40 nM T13201 C7T1ZF 10788101 Ki = 290 nM T13201 C3P7LZ 10792025 Ki = 180 nM T13201 CDO17N 10792606 Ki = 305000 nM T13201 C5Q0HP 10792608 Ki = 130000 nM T13201 CCF8T2 10792692 Ki = 360 nM T13201 CMY20D 10792820 Ki = 10 nM T13201 CR9A3S 10792923 Ki = 610 nM T13201 CCYS21 10793062 Ki = 24 nM T13201 CK5ZL2 10793077 Ki = 1450 nM T13201 CHD5Q2 10793387 Ki = 550 nM T13201 CX0BW6 10793389 Ki = 11 nM T13201 CEY35S 10793458 Ki = 600 nM T13201 CFL4G8 10800492 Ki = 540 nM T13201 CH1F0I 10803110 Ki = 23500 nM T13201 C25VZF 10804238 Ki = 25200 nM T13201 CU1BS8 10804376 Ki = 20000 nM T13201 CGY6S7 10804696 Ki = 600 nM T13201 C7N2LO 10805708 Ki = 20000 nM T13201 C1QF3B 10806893 Ki = 620 nM T13201 CH1A4N 10807238 Ki = 10 nM T13201 CC0V8S 10808608 Ki = 55 nM T13201 CU9F7V 10810684 Ki > 200 nM T13201 CJGV81 10810883 Ki = 51 nM T13201 C58LOZ 10812489 Ki = 610 nM T13201 C42JTI 10813047 Ki = 55 nM T13201 CQR74O 10813858 Ki = 3000 nM T13201 C4Q1BT 10814610 Ki = 1500 nM T13201 CPG8X7 10815580 Ki = 1350 nM T13201 CIU0T4 10815639 Ki = 800 nM T13201 C9S1KI 10816020 Ki = 42000 nM T13201 CZ8SC0 10816485 Ki = 1500 nM T13201 CDX47C 10817418 Ki = 5100 nM T13201 CPU04C 10817804 Ki = 1000 nM T13201 CI21MQ 10817828 Ki = 15000 nM T13201 CW4J0M 10817935 Ki = 380 nM T13201 CR6WQ9 10818727 Ki = 810 nM T13201 CQBR40 10825041 Ki = 965 nM T13201 CVN37O 10825297 Ki = 500 nM T13201 CW9YL5 10827620 Ki = 320 nM T13201 CIW28L 10829558 Ki = 550 nM T13201 CHE35M 10832570 Ki = 525 nM T13201 C3TN8I 10832697 Ki = 1400 nM T13201 CA13RM 10833200 Ki = 250 nM T13201 COE82D 10833334 Ki = 10 nM T13201 CQM97L 10833411 Ki = 520 nM T13201 CMI8K1 10833817 Ki = 3000 nM T13201 C9M1JI 10834357 Ki > 200 nM T13201 C6U5RE 10834502 Ki = 1250 nM T13201 C1R4OZ 10836567 Ki = 500 nM T13201 CWF8K2 10836730 Ki = 75 nM T13201 CLS5J3 10836786 Ki = 7000 nM T13201 C0IY7D 10836837 Ki = 45 nM T13201 C3NIE1 10836973 Ki = 20 nM T13201 CO6C3T 10837292 Ki = 500 nM T13201 CR0E9Q 10837740 Ki = 105 nM T13201 C3XU6W 10838049 Ki = 450 nM T13201 C32QME 10838459 Ki = 2000 nM T13201 C2P7QW 10839526 Ki = 700 nM T13201 CBE3L7 10839725 Ki = 6600 nM T13201 CLIK46 10840741 Ki = 34000 nM T13201 CM4ZJ7 10841903 Ki = 950 nM T13201 CX9B7K 10841917 Ki = 20000 nM T13201 CJI5F0 10841980 Ki = 2300 nM T13201 CWVN58 10842131 Ki = 350 nM T13201 CG6XO9 10842189 Ki = 1450 nM T13201 CMA41F 10842208 Ki = 45 nM T13201 C93MDS 10842492 Ki = 50 nM T13201 C98LNY 10842547 Ki = 14 nM T13201 C5Z3AD 10842801 Ki = 17 nM T13201 C3W8OJ 10842917 Ki = 3000 nM T13201 CW28MA 10843175 Ki = 1100 nM T13201 CB2KJ7 10847811 Ki = 1400 nM T13201 CO2SP9 10847812 Ki = 15000 nM T13201 CQ0HY2 10848746 Ki = 850 nM T13201 CMH6X5 10850981 Ki = 62 nM T13201 C06ORC 10851952 Ki = 510 nM T13201 C98OIB 10852025 Ki = 540 nM T13201 CH0A6S 10852944 Ki = 1040 nM T13201 CF9SV4 10861185 Ki = 62 nM T13201 CZ4P8F 10862789 Ki = 550 nM T13201 C1B2IY 10863970 Ki = 1.6 nM T13201 C19MNG 10864178 Ki = 12500 nM T13201 CPN13K 10864662 Ki = 510 nM T13201 CY82EF 10865353 Ki = 5600 nM T13201 C4E8SG 10865419 Ki = 105 nM T13201 C8M4QY 10865548 Ki = 3800 nM T13201 C8OKX5 10865717 Ki = 25 nM T13201 C7DV4E 10868086 Ki = 43 nM T13201 CQN7G6 10869299 Ki = 3900 nM T13201 CP8DF6 10871235 Ki = 20500 nM T13201 CUKT63 10872446 Ki = 1100 nM T13201 CB3U9M 10874216 Ki = 2.1 nM T13201 C8TM4D 10875038 Ki = 245 nM T13201 C4CM8X 10875810 Ki = 78 nM T13201 CG0Z6I 10876077 Ki = 250 nM T13201 CFXH68 10876514 Ki = 36 nM T13201 CT0KQ8 10878827 Ki = 3800 nM T13201 C0M3OP 10881177 Ki = 1260 nM T13201 CWKM78 10884587 Ki = 405 nM T13201 C23JVY 10886478 Ki = 210 nM T13201 C1YK9S 10886620 Ki = 120 nM T13201 C6YGB0 10886642 Ki = 41 nM T13201 CO0V5G 10887065 Ki = 9500 nM T13201 C1LX6K 10887220 Ki = 155 nM T13201 CN2L6A 10891750 Ki = 415 nM T13201 CH3LK7 10893334 Ki = 50 nM T13201 CR81KU 10895699 Ki = 225 nM T13201 CY9O1Q 10895884 Ki = 360 nM T13201 CKL08U 10897133 Ki = 360 nM T13201 CBNU79 10897483 Ki = 460 nM T13201 CC51VX 10898100 Ki = 21 nM T13201 C9C5HV 10898245 Ki = 15 nM T13201 CCW0R7 10899319 Ki = 252 nM T13201 C2MY5U 10904482 Ki = 30500 nM T13201 CX2K9L 10904983 Ki = 960 nM T13201 C7SH5U 10905170 Ki = 56 nM T13201 CWGB92 10907843 Ki = 550 nM T13201 C2VEZ9 10907925 Ki = 52 nM T13201 C90ZUF 10908674 Ki = 55 nM T13201 CIO06R 10915496 Ki = 900 nM T13201 C0BP2F 10915515 Ki = 610 nM T13201 CG10IV 10916112 Ki = 46 nM T13201 C3WOS1 10917392 Ki = 2600 nM T13201 CUEX85 10918009 Ki = 345 nM T13201 C50OCY 10918511 Ki = 7450 nM T13201 C8RXZ0 10919029 Ki = 33 nM T13201 C6EPH9 10919571 Ki = 578 nM T13201 CP2Z4G 10919976 Ki = 89 nM T13201 CTDR05 10920174 Ki = 43 nM T13201 C8CV1Z 10923837 Ki = 454 nM T13201 C8TSL7 10926221 Ki = 275 nM T13201 CL5D1P 10926842 Ki = 415000 nM T13201 CVR31W 10930187 Ki = 96 nM T13201 C3WN6P 10931938 Ki = 401 nM T13201 C7FP4E 10932133 Ki = 0.88 nM T13201 CGI4X1 10933094 Ki > 10000 nM T13201 CHZI28 10935067 Ki = 23000 nM T13201 C8FIB7 10935528 Ki = 32700 nM T13201 CD3GB7 10937101 Ki = 3.1 nM T13201 CO17LZ 10948175 Ki = 410 nM T13201 C8P1ER 10950587 Ki = 300 nM T13201 CZA48D 10952342 Ki = 30 nM T13201 CPC86B 10952559 Ki = 6150 nM T13201 CZAG71 10952780 Ki = 125 nM T13201 CW2K3M 10953423 Ki = 200000 nM T13201 CN27BY 10953838 Ki > 100000 nM T13201 C3F9WR 10957702 Ki = 1300 nM T13201 CIXO05 10959593 Ki = 2.5 nM T13201 CVG71F 10961747 Ki = 650 nM T13201 CEV7Z1 10962037 Ki = 1 nM T13201 CQO1E7 10962986 Ki = 2.1 nM T13201 C5ZPE9 10963315 Ki = 30 nM T13201 C0K1QF 10963422 Ki = 225 nM T13201 C4B5DJ 10963712 Ki = 300 nM T13201 C9NC5T 10964817 IC50 = 113000000 nM T13201 CCV07P 10970019 Ki = 25800 nM T13201 CG08QZ 10970428 Ki = 1200 nM T13201 C1H7KL 10970502 Ki = 1000 nM T13201 CZPG31 10972292 Ki = 250 nM T13201 C3IDH7 10974944 Ki = 79 nM T13201 CU4TO5 10979790 Ki = 710 nM T13201 CFL46Z 10980153 Ki = 70 nM T13201 C40UVN 10980851 Ki = 1760 nM T13201 C59AQM 10983522 Ki = 215 nM T13201 C73HZT 10983658 Ki = 1.7 nM T13201 CM6Z2B 10983679 Ki = 700 nM T13201 C4MXZ2 10985404 Ki = 33 nM T13201 CG61PD 10994426 Ki = 290 nM T13201 CP5A7X 10995068 Ki = 4000 nM T13201 CE23PC 10995136 Ki = 1.9 nM T13201 C6VG2U 10995156 Ki = 54 nM T13201 C69NOP 10995214 Ki = 12500 nM T13201 COQ4Y6 10995233 Ki = 210 nM T13201 CU91KW 10995327 Ki = 430 nM T13201 C7X4SM 10995402 Ki = 47 nM T13201 C91OEI 10995928 Ki = 76 nM T13201 C8JAX5 10996222 Ki = 9800 nM T13201 CIO7M2 10996308 Ki = 150 nM T13201 C60TSD 10996432 Ki = 16 nM T13201 CCIT95 11003980 Ki = 1.1 nM T13201 C0R1IV 11004960 Ki = 430 nM T13201 C8YZ0I 11005191 Ki = 510 nM T13201 CVYW37 11006065 Ki = 1050 nM T13201 C7WEZ4 11009332 Ki = 72000 nM T13201 C1D7XA 11011569 Ki = 7600 nM T13201 C9IF1C 11013393 Ki = 432 nM T13201 CEY2A4 11014189 Ki = 3300 nM T13201 CD4JQ1 11015176 Ki = 1.9 nM T13201 C2Y6HS 11016006 Ki = 850 nM T13201 CH47PL 11016833 Ki = 200 nM T13201 CNCX57 11017060 Ki = 7200 nM T13201 CDR0Y6 11017072 Ki = 39 nM T13201 C69TDE 11017073 Ki = 610 nM T13201 C4WU6R 11017835 Ki = 79 nM T13201 C8VI2F 11018004 Ki = 350 nM T13201 C2G5AL 11018133 Ki = 105 nM T13201 CX1F7U 11018241 Ki = 25 nM T13201 C9L3MK 11018318 Ki = 85 nM T13201 CC0F9X 11018319 Ki = 76 nM T13201 C6UD9P 11018463 Ki = 76 nM T13201 CAED68 11021701 Ki = 415 nM T13201 CLV4S2 11024707 Ki = 50 nM T13201 CDB16V 11026415 Ki = 1 nM T13201 C5CJU7 11028005 Ki = 8600 nM T13201 CLM10Q 11028999 Ki = 135 nM T13201 CD8HS3 11031678 Ki = 37 nM T13201 CWO84N 11032771 Ki = 115 nM T13201 CLN35C 11034434 Ki = 1000 nM T13201 C36BAC 11034581 Ki > 100000 nM T13201 CFBO12 11035956 Ki = 520 nM T13201 CN6QX1 11036198 Ki = 12500 nM T13201 CB4M2O 11036993 Ki = 240 nM T13201 COA8S5 11039158 Ki = 200 nM T13201 CL46GE 11039314 Ki = 32 nM T13201 CA1P7Q 11045484 Ki = 975 nM T13201 CV75NH 11047521 Ki = 5.7 nM T13201 CJ3WY1 11048561 Ki = 9200 nM T13201 CVW8K3 11048831 Ki = 16000 nM T13201 CC6K7Q 11055293 Ki = 21300 nM T13201 COWY75 11055630 Ki = 19000 nM T13201 CJ2M4S 11055723 Ki = 3600 nM T13201 CO2F4K 11058711 Ki = 800 nM T13201 C3ZP6U 11058734 Ki = 515 nM T13201 CFU60B 11060209 Ki = 48 nM T13201 CC7X2Z 11060668 Ki = 500 nM T13201 CT2D9I 11060771 Ki = 12000 nM T13201 C6FA8Y 11060833 Ki = 62 nM T13201 C5X4DW 11060882 Ki = 290 nM T13201 CQBP46 11061197 Ki = 438 nM T13201 C1C4OI 11061783 Ki = 160 nM T13201 CP1U3L 11062054 Ki = 49 nM T13201 C36YHJ 11067477 Ki = 13000 nM T13201 C8C6ER 11069133 Ki = 1.4 nM T13201 CWM7C8 11071324 Ki = 11500 nM T13201 CU5NJ9 11071502 Ki = 21000 nM T13201 CRL5I3 11072036 Ki = 130 nM T13201 COGV98 11074431 Ki > 20000 nM T13201 C1BAR9 11077028 Ki = 27000 nM T13201 CYT4G0 11078481 Ki = 1020 nM T13201 CMQ2Y8 11079355 Ki = 600 nM T13201 CJW7Z3 11081263 Ki = 640 nM T13201 CWTS45 11081678 Ki = 43 nM T13201 CASO94 11081987 Ki = 1200 nM T13201 CIC47S 11082122 Ki = 760 nM T13201 C6WU3G 11082240 Ki = 66 nM T13201 C2NXV7 11082357 Ki = 230 nM T13201 CIAW06 11082579 Ki = 36 nM T13201 C3O5JB 11083515 Ki = 16 nM T13201 C9YZA3 11089252 Ki = 23000 nM T13201 CEM9W0 11091166 Ki = 268 nM T13201 CHA42C 11092653 Ki = 945 nM T13201 CS8W3K 11092704 Ki = 8900 nM T13201 CSL53A 11093007 Ki = 123 nM T13201 CYST27 11093710 Ki = 58 nM T13201 CMK4Y0 11096006 Ki = 1289 nM T13201 C2P8ZU 11099090 Ki = 3450 nM T13201 CKF5V1 11099458 Ki = 3500 nM T13201 C14ZGJ 11101626 Ki = 380 nM T13201 C8DOK1 11102362 Ki = 44 nM T13201 C7RZW3 11103137 Ki = 5.2 nM T13201 COJU46 11103269 Ki = 10000 nM T13201 CJF79N 11103375 Ki = 130 nM T13201 CK12PR 11103476 Ki = 250 nM T13201 CWB10K 11103986 Ki = 9 nM T13201 C53LWS 11104965 Ki = 50 nM T13201 CZ91PR 11109866 Ki = 1200 nM T13201 CYI5F6 11110737 Ki = 20600 nM T13201 CVZ89X 11112315 Ki = 273000 nM T13201 CSI1G6 11114605 Ki = 39 nM T13201 CV8S7A 11114620 Ki = 175 nM T13201 C4CE8S 11114939 Ki = 93 nM T13201 CDY1T6 11115104 Ki = 50 nM T13201 CYQ01S 11115351 Ki = 9.5 nM T13201 CH6IE3 11117198 Ki = 39.6 nM T13201 C9UJ8I 11125027 Ki = 240 nM T13201 C31VGI 11125411 Ki = 37 nM T13201 C8X2DC 11127784 Ki = 69.9 nM T13201 C6RM4H 11134231 Ki = 5 nM T13201 CU8OF2 11141517 Ki = 35600 nM T13201 CZ09RJ 11143896 Ki = 48 nM T13201 CC28PQ 11144024 Ki = 14660 nM T13201 CG36VZ 11144533 Ki = 43 nM T13201 C25CRH 11146161 Ki = 180 nM T13201 CO6X8J 11147037 Ki = 54 nM T13201 C5WS3E 11147931 IC50 = 8810 nM T13201 CP3CU4 11157709 Ki = 3 nM T13201 CC4IE1 11158128 Ki = 4 nM T13201 CPB0A5 11164855 Ki = 760 nM T13201 CEYJ94 11165541 Ki = 580 nM T13201 C50HJY 11177131 Ki = 1150 nM T13201 C3PJ6O 11177505 Ki = 1300 nM T13201 CIL4M9 11183499 Ki > 100000 nM T13201 C39IDU 11183936 Ki = 13440 nM T13201 C4W0YX 11186322 Ki = 58000 nM T13201 C31DIQ 11188711 Ki = 4800 nM T13201 C5C6MG 11194613 Ki = 4620 nM T13201 C5Y1CV 11196316 Ki > 1000000 nM T13201 C75FMT 11199252 Ki = 980 nM T13201 CFG37K 11209006 Ki = 14 nM T13201 C0P8JA 11215523 Ki = 950 nM T13201 C2AFO0 11216333 Ki = 630 nM T13201 C5L7NR 11217340 Ki = 990000 nM T13201 CJOR84 11220854 Ki = 510 nM T13201 CY2VA5 11221764 Ki = 1500 nM T13201 CY1P4Q 11223689 Ki = 865 nM T13201 CY9W5K 11226359 Ki = 6000 nM T13201 C39QJA 11234047 Ki = 270 nM T13201 CXAS45 11235150 Ki = 1200 nM T13201 C8O1FM 11239393 Ki = 6 nM T13201 CHC42Y 11245700 Ki = 3600 nM T13201 C92XHG 11245995 Ki = 1750 nM T13201 CGE40M 11245996 Ki = 950 nM T13201 CCLV87 11247335 Ki = 1450 nM T13201 CN86YV 11250791 Ki = 5 nM T13201 CI7YT0 11252120 Ki = 3100 nM T13201 C7UVW8 11258440 Ki = 700 nM T13201 C12URI 11261582 Ki = 4 nM T13201 CIR6A0 11262484 Ki = 10 nM T13201 CV7T2K 11269105 Ki = 1300 nM T13201 C5P7KN 11269273 Ki = 270 nM T13201 C43WCH 11269442 Ki = 1000 nM T13201 C7FA3C 11274029 Ki = 12 nM T13201 CF1ZC0 11278507 Ki = 374000 nM T13201 CCSA87 11280465 Ki = 318 nM T13201 CF15AS 11287957 Ki > 10000 nM T13201 CG28LP 11290362 Ki = 239000 nM T13201 C0H6GB 11292444 Ki = 860 nM T13201 C1FJ7I 11304583 Ki = 4900 nM T13201 C3CDO1 11309586 Ki = 687 nM T13201 CRP08M 11310883 IC50 = 5310 nM T13201 CBC47W 11312414 Ki = 150 nM T13201 CAU4B5 11317320 Ki = 2400 nM T13201 CB4U3M 11318985 Ki = 1500 nM T13201 CHA0V5 11321514 Ki = 830 nM T13201 CDLR79 11321711 Ki = 19 nM T13201 CA6T0Z 11322287 Ki = 12630 nM T13201 C8ZA1X 11326347 Ki = 900 nM T13201 C84HMR 11329414 Ki = 740 nM T13201 CU73JN 11339017 Ki = 600 nM T13201 C8Q5VJ 11342941 Ki = 8 nM T13201 CV80KU 11346010 Ki = 7500 nM T13201 CCY4G5 11350445 Ki = 4700 nM T13201 CDLS49 11350634 Ki = 930 nM T13201 C3NGH2 11352609 Ki = 6300 nM T13201 C8PM3Z 11353795 Ki = 1300 nM T13201 C8MI3Z 11361075 Ki = 1080 nM T13201 C27RAM 11361542 Ki = 760 nM T13201 CY3B6F 11362509 Ki = 3600 nM T13201 CM8Y1J 11367571 IC50 = 6710 nM T13201 CM1XU5 11373291 Ki = 800 nM T13201 C6QO0H 11384370 Ki = 750 nM T13201 CY64KU 11385765 Ki = 0.6 nM T13201 CIQ5K7 11387799 Ki = 7 nM T13201 C7MK2E 11390955 Ki = 3540 nM T13201 CVT2K6 11396353 Ki = 550 nM T13201 CT3E0Y 11399060 Ki = 980 nM T13201 C6RUJ7 11399350 Ki = 3 nM T13201 CEO47P 11399506 Ki = 1100 nM T13201 CH98MP 11399715 Ki = 5 nM T13201 CBVL07 11407223 Ki = 1160 nM T13201 C3KV6R 11407281 Ki = 3400 nM T13201 C8DF5O 11416806 Ki = 65000 nM T13201 CG1A5D 11427826 Ki = 5100 nM T13201 CGPE75 11428235 Ki = 250 nM T13201 CT3NI0 11433608 Ki = 4 nM T13201 C3KRG4 11433767 Ki = 9 nM T13201 CK7D5V 11438030 Ki = 201000 nM T13201 CUR65I 11441308 Ki = 78 nM T13201 CTU87D 11441601 Ki = 1360 nM T13201 C7EOG0 11441729 Ki = 1870 nM T13201 C41CHM 11445520 Ki = 480 nM T13201 CMS0Q5 11445529 Ki = 5 nM T13201 C32QDC 11453942 Ki = 1960 nM T13201 C54AMO 11454377 Ki = 320 nM T13201 C4BQM5 11455128 Ki = 6100 nM T13201 C2J9BG 11463026 Ki = 1450 nM T13201 CFER43 11467281 Ki = 1450 nM T13201 CM9I6W 11467962 Ki = 5 nM T13201 CQ1D6E 11470070 IC50 = 7360 nM T13201 CNM06W 11475346 Ki = 940 nM T13201 C91XWJ 11478542 Ki = 1400 nM T13201 CIWG06 11479385 Ki = 6 nM T13201 CCY54I 11479559 Ki = 8 nM T13201 C0WCE4 11482579 Ki = 428000 nM T13201 CL1RC2 11485376 Ki = 760 nM T13201 CQ9H8J 11490915 Ki = 1070 nM T13201 C8YO5G 11508929 Ki = 14700 nM T13201 CNFY48 11514219 Ki = 97 nM T13201 CU8YH7 11533895 Ki = 32 nM T13201 CP8AX2 11540662 Ki = 8.6 nM T13201 CJZ9N8 11573504 Ki = 12300 nM T13201 CIMD40 11578176 Ki = 5530 nM T13201 CXB86F 11579563 Ki = 12130 nM T13201 CUJI91 11581618 Ki = 10000 nM T13201 CT7LD4 11588141 Ki = 541 nM T13201 CDS25O 11593765 IC50 = 1600 nM T13201 CCB82K 11596108 Ki = 96 nM T13201 C3FJQ8 11602375 Ki = 307000 nM T13201 C9QL2F 11615432 Ki = 3406 nM T13201 C36MZP 11616716 Ki = 104 nM T13201 CK38DO 11624852 Ki = 700 nM T13201 CV02TF 11632228 Ki = 338 nM T13201 CDU79V 11637531 Ki = 14210 nM T13201 C4EC3U 11663528 Ki = 32000 nM T13201 C95PYS 11667431 Ki = 3 nM T13201 C9JR2I 11674590 Ki = 44100 nM T13201 CRG49U 11674754 Ki = 138 nM T13201 CPGO32 11675510 Ki = 7000 nM T13201 C7ZPR9 11681852 Ki = 75 nM T13201 C8F0SQ 11687376 IC50 = 25000 nM T13201 CCG17H 11688636 Ki = 63 nM T13201 CF8IT6 11696964 Ki = 3 nM T13201 CX4W3J 11701693 Ki = 12320 nM T13201 C4VZO5 11709992 Ki = 116 nM T13201 CHAN30 11714982 Ki = 37 nM T13201 C5QIK4 11721174 Ki = 280000 nM T13201 C1G0JC 11727638 Ki = 65 nM T13201 CB0EA2 11727760 Ki = 780 nM T13201 CWV01J 11728049 Ki = 1540 nM T13201 CJXL89 11728811 Ki = 45 nM T13201 CO03JM 11729079 Ki = 50 nM T13201 CD16NH 11729087 Ki = 400 nM T13201 C0L3RF 11729108 Ki = 62 nM T13201 CV6LK7 11729550 Ki = 620 nM T13201 CYI4S1 11729993 Ki = 970 nM T13201 CH7BF3 11731156 Ki = 450 nM T13201 CE14NA 11731409 Ki = 290 nM T13201 CAW47S 11733056 Ki = 1.3 nM T13201 CEGC64 11735346 Ki = 290 nM T13201 C5YD7H 11735447 Ki = 23 nM T13201 CB93NJ 11738933 Ki = 231000 nM T13201 C4FA0T 11740604 Ki = 18 nM T13201 C2D6WI 11748537 Ki = 23000 nM T13201 C0TFH3 11760610 Ki = 360 nM T13201 CX5LA8 11763331 Ki = 4100 nM T13201 CP78CU 11763512 Ki = 11 nM T13201 CBN39F 11767393 Ki = 240 nM T13201 CWM5I6 11773896 Ki = 1250 nM T13201 CV68TJ 11774586 Ki = 1300 nM T13201 CH7Q5S 11777250 Ki > 10000 nM T13201 C98EGL 11782389 Ki = 1300 nM T13201 C9J0YH 11782553 Ki = 950 nM T13201 CJ35OU 11782715 Ki = 250 nM T13201 C37CKB 11782720 Ki = 105 nM T13201 C28PBF 11782912 Ki = 21800 nM T13201 CC9L1G 11783323 Ki = 3500 nM T13201 C6S8WR 11786209 Ki = 3 nM T13201 C4BH9A 11788388 Ki = 800000 nM T13201 C7BV5P 11792968 Ki = 8 nM T13201 C4U8QN 11794109 Ki = 30 nM T13201 CW32BE 11794202 Ki = 1200 nM T13201 CV7HN1 11795548 Ki = 4000 nM T13201 CT2G8Q 11796369 Ki = 710 nM T13201 CG6Z5X 11797062 Ki = 32000 nM T13201 C19RCP 11799753 Ki > 200 nM T13201 C07QLV 11800828 Ki = 15000 nM T13201 C8X0GK 11800862 Ki = 11 nM T13201 CE1S6W 11801129 Ki = 400 nM T13201 C3E7CX 11801767 Ki = 41 nM T13201 CNB5F6 11802420 Ki = 11 nM T13201 CLC27W 11802422 Ki = 1140 nM T13201 C93PTE 11802889 Ki = 53 nM T13201 CH7OA8 11803531 Ki = 800 nM T13201 CSD5K9 11806775 Ki = 369 nM T13201 CL69XF 11809670 Ki = 12000 nM T13201 C95JYR 11813616 Ki = 870 nM T13201 C45XIB 11814933 Ki = 65 nM T13201 C0RZ9Y 11816502 Ki = 410 nM T13201 C8DY3Z 11817193 IC50 = 8020 nM T13201 C73SVE 11817275 Ki = 73.5 nM T13201 CTR0U7 11823783 Ki = 7800 nM T13201 C9CJU1 11824513 Ki = 1000 nM T13201 C0VWS3 11824695 Ki = 280 nM T13201 CO7K8V 11826660 Ki = 900 nM T13201 C1DB0Z 11828379 Ki = 220 nM T13201 C0OD9Y 11828467 Ki = 450 nM T13201 C18JIA 11828627 Ki = 5400 nM T13201 CIWV68 11828670 Ki = 335 nM T13201 CE71FU 11828964 Ki = 102 nM T13201 C0CR2G 11848185 Ki = 100 nM T13201 C45NRP 11851425 Ki = 5800 nM T13201 CJRD82 11966600 Ki = 110 nM T13201 C4T8BS 11967023 Ki = 155 nM T13201 CXSE37 11967046 Ki = 325 nM T13201 C9VM6I 11967472 Ki = 70 nM T13201 CQXG94 11970596 Ki = 9400 nM T13201 CZD0B3 11974341 Ki = 5600 nM T13201 C27HSO 11974343 Ki = 10400 nM T13201 CCM17V 11974451 Ki = 6600 nM T13201 CX4IJ0 11974452 Ki = 9100 nM T13201 C59UEI 11974453 Ki = 9500 nM T13201 CYS7X0 11974454 Ki = 9300 nM T13201 C09JGZ 11974455 Ki = 3600 nM T13201 CS9VL2 11974456 Ki = 5100 nM T13201 CP39YI 11974558 Ki = 5400 nM T13201 CB97SM 11974559 Ki = 3400 nM T13201 CE8WN6 11974560 Ki = 5800 nM T13201 C06CBY 11974561 Ki = 4800 nM T13201 CU6K0N 11974562 Ki = 3500 nM T13201 CI7OE1 11974563 Ki = 8700 nM T13201 C6Z5DX 11974630 Ki = 1200 nM T13201 CW4X9G 11974631 Ki = 9200 nM T13201 CEBO65 11974632 Ki = 2300 nM T13201 CGQ6B7 11974724 Ki = 3900 nM T13201 CHO9T1 11974725 Ki = 2000 nM T13201 CC8TS1 11974727 Ki = 2400 nM T13201 CDL18J 11974728 Ki = 4400 nM T13201 C7G3YS 11974830 Ki = 9.6 nM T13201 C1C4JW 11974831 Ki = 3100 nM T13201 CXW89D 12004261 Ki = 85 nM T13201 C0L4OC 12049163 Ki > 100000 nM T13201 C4ZYQ1 12049713 Ki = 1270000 nM T13201 CNHD71 12051191 Ki > 200000 nM T13201 CMPA32 12066940 Ki > 500000 nM T13201 CB15KR 12066941 Ki > 500000 nM T13201 C2XBZ3 12070806 Ki = 280 nM T13201 C32TWU 12094253 Ki = 26.6 nM T13201 CREV05 12140130 Ki = 13250 nM T13201 C6P1VC 12188108 Ki > 10000 nM T13201 C3C9ON 12226066 Ki = 30300 nM T13201 CCY51E 12237458 Ki > 10000 nM T13201 C60EFT 12354987 Ki = 130 nM T13201 CPU03D 12355589 Ki = 173 nM T13201 CSYD70 12355590 Ki = 164 nM T13201 C18LXJ 12411101 Ki = 3.8 nM T13201 C0C8FG 12411107 Ki = 113 nM T13201 C5NK2I 12420669 IC50 = 9850 nM T13201 C0JID3 12447203 Ki = 12000 nM T13201 CLB1E3 12499681 Ki > 10000 nM T13201 CP87GR 12516475 Ki = 32.9 nM T13201 C5RS4H 12528487 Ki = 968.7 nM T13201 CM8TP6 12528490 Ki = 3809 nM T13201 C35CMO 12589789 Ki > 10000 nM T13201 CTHQ39 12635073 Ki = 68000 nM T13201 CIQX87 12635074 Ki = 15000 nM T13201 CK90BP 12765315 Ki = 6640 nM T13201 CZCF65 12914626 Ki = 40000 nM T13201 C1GNM5 12914627 Ki = 3700 nM T13201 CO8WC5 12938307 Ki = 263 nM T13201 CP70LE 12954894 Ki = 371 nM T13201 C4IKA3 13087489 Ki = 401 nM T13201 CF2BM7 13177311 Ki = 332 nM T13201 C8VM1A 13201770 Ki = 390 nM T13201 CI31SL 13204988 Ki = 4060 nM T13201 CV1UF4 13306723 Ki = 13.1 nM T13201 C85GSD 13360355 Ki = 7800 nM T13201 CX7M9C 13373975 Ki > 10000 nM T13201 CHC41Q 13381193 Ki > 10000 nM T13201 COLK69 13419352 Ki > 10000 nM T13201 CSN63J 13427336 IC50 = 11240 nM T13201 C3HOK8 13580495 Ki = 59000 nM T13201 CFN29Y 13584466 Ki > 10000 nM T13201 CQTX49 13738810 IC50 = 5932 nM T13201 C57SFI 13801611 Ki > 100000 nM T13201 C24OQJ 13803658 IC50 = 4810 nM T13201 CC25BI 13927398 Ki = 85000 nM T13201 CTYP72 13949092 Ki > 10000 nM T13201 CR6HB5 13949095 Ki > 10000 nM T13201 CFMK94 13949102 Ki > 10000 nM T13201 C7K4JV 14024589 Ki = 6857 nM T13201 C4UG2O 14057643 Ki = 5840 nM T13201 CLS53V 14151811 IC50 > 10000 nM T13201 CQ3D9C 14151815 IC50 > 10000 nM T13201 CNZ6H2 14205726 Ki > 300000000 nM T13201 CA5Q3H 14425149 Ki = 200.5 nM T13201 CXYO59 14435742 IC50 = 8370 nM T13201 C92OEB 14498136 Ki = 40.4 nM T13201 CHOG93 14611919 Ki = 7.5 nM T13201 CZ6SN8 14777102 Ki = 337 nM T13201 C76ASY 14787919 Ki > 200000 nM T13201 C35DGV 14873166 Ki > 10000 nM T13201 C9CLH4 14873170 Ki > 10000 nM T13201 C9K0LX 14873174 Ki > 10000 nM T13201 CM34ER 14873177 Ki > 10000 nM T13201 CH5YR2 15014351 Ki > 200000 nM T13201 CW3X5A 15038375 Ki = 237000 nM T13201 C7XD2T 15118768 Ki = 8460 nM T13201 CX26PT 15219881 Ki = 16 nM T13201 CK8GE9 15230629 Ki = 1920 nM T13201 C6F3GK 15267134 Ki = 247.23 nM T13201 CDE4F9 15290967 Ki > 10000 nM T13201 C1IZ7D 15296597 Ki = 195 nM T13201 CJ7V8G 15381187 Ki = 641 nM T13201 C9X6AG 15381192 Ki = 612 nM T13201 CW72MS 15438999 Ki > 50000 nM T13201 C7R5AH 15476112 Ki = 6180 nM T13201 C3CTS0 15523879 Ki = 55.4 nM T13201 CFC2E0 15546406 Ki = 30 nM T13201 C2G4FH 15599374 Ki = 982 nM T13201 CT73PL 15618966 Ki = 1150 nM T13201 CLIO60 15645619 Ki = 378.6 nM T13201 C8PMQ9 15729847 Ki = 4690 nM T13201 CLT47Z 15783680 Ki > 10000 nM T13201 C6VR7G 15815634 Ki = 85000 nM T13201 C6F0XZ 15818962 Ki > 10000 nM T13201 C8PER5 15938557 Ki > 500000 nM T13201 C3W2MB 15939939 Ki > 10000 nM T13201 CB3S7I 16007202 Ki = 59 nM T13201 CM06OZ 16046226 Ki = 2600 nM T13201 CVZG29 16072592 Ki = 3600 nM T13201 CB73ST 16072595 Ki = 1850 nM T13201 C6U0VS 16078349 Ki = 62 nM T13201 CUT32D 16078350 Ki > 1000 nM T13201 C4JIO0 16078351 Ki = 30 nM T13201 C23FGI 16078837 Ki > 100000 nM T13201 CQ0UX9 16082752 Ki = 97 nM T13201 CBRL45 16082753 Ki = 71 nM T13201 C0BIQ3 16082754 Ki = 60 nM T13201 C6KN4Z 16082755 Ki = 41 nM T13201 C94FZV 16082756 Ki = 69 nM T13201 C85HIK 16082757 Ki = 5115 nM T13201 CC74NH 16087011 Ki > 10000 nM T13201 C1CD5B 16087012 Ki > 10000 nM T13201 C8AP5W 16087015 Ki > 10000 nM T13201 CLNI97 16087025 Ki > 10000 nM T13201 CBWD20 16087028 Ki > 10000 nM T13201 CN1XR0 16087029 Ki > 10000 nM T13201 C3GMJ8 16087031 Ki > 10000 nM T13201 CC0Z4V 16119626 Ki = 3870 nM T13201 CB7CU4 16122563 Ki = 1200 nM T13201 CV5O8W 16125524 Ki = 7 nM T13201 CZ7T4C 16125526 Ki = 1500 nM T13201 CS78TE 16125527 Ki = 6.9 nM T13201 C1Z9GQ 16125580 Ki = 8.1 nM T13201 CE4SB2 16125581 Ki = 4700 nM T13201 CWM0L9 16125582 Ki = 4400 nM T13201 C4SD3N 16125583 Ki = 7.3 nM T13201 CPU0F5 16219477 Ki = 7610 nM T13201 CA6VB3 16221528 Ki = 10700 nM T13201 CQGZ56 16221529 Ki = 11400 nM T13201 C79XIS 16221532 Ki = 11200 nM T13201 CPD68G 16221533 Ki = 11900 nM T13201 CPR94Q 16221534 Ki = 158000 nM T13201 CZO0W5 16221535 Ki = 10500 nM T13201 C0UO9G 16221580 Ki = 9600 nM T13201 CN03IT 16227153 Ki = 192 nM T13201 CGB45O 16235229 Ki = 374 nM T13201 CV35UO 16450309 IC50 = 95700 nM T13201 CG7OL3 16693908 Ki = 52400000 nM T13201 CMB87O 16717602 Ki > 10000 nM T13201 COQU32 16729004 Ki = 873 nM T13201 CTK68M 17249579 Ki = 9.8 nM T13201 C5DT7E 17250082 Ki = 436 nM T13201 C6THW2 17268490 Ki = 4330 nM T13201 C5CE8Z 17371280 Ki = 39.6 nM T13201 CA4OE9 17371576 Ki = 58.9 nM T13201 C73YML 17385730 Ki = 324 nM T13201 C91LAN 17413757 Ki = 1980 nM T13201 C5M9DR 17433209 Ki > 10000 nM T13201 CYLM41 17492191 Ki > 10000 nM T13201 CDWU20 17537594 Ki = 8.9 nM T13201 CUP95O 17562622 Ki = 186.6 nM T13201 CK7D2I 17748220 Ki = 11000 nM T13201 CLY1N4 17757567 Ki = 8840 nM T13201 CVN21Y 17770844 Ki = 10830 nM T13201 C3AX8E 17774014 Ki = 491 nM T13201 C6SFI8 18268734 Ki = 6331 nM T13201 CR9VF3 18668331 Ki = 785 nM T13201 CQE5K4 18710120 Ki > 200000 nM T13201 C60NAV 18971452 Ki = 453 nM T13201 C6HO7T 18990081 Ki = 266 nM T13201 C2K5BX 19374444 Ki = 762 nM T13201 CIEH93 19382975 IC50 > 10000 nM T13201 C97MSK 19782950 Ki > 100000 nM T13201 C62PKT 19838794 Ki = 50.1 nM T13201 CU3QS7 19898674 Ki > 10000 nM T13201 CB46JX 20109894 Ki = 42 nM T13201 CGE35Q 20182298 Ki = 5.3 nM T13201 CDU40W 20184392 Ki = 24900 nM T13201 CXJ2H4 20195196 Ki > 100000 nM T13201 C8Z1CM 20216502 Ki = 710 nM T13201 C1H6GV 20360268 Ki > 100000 nM T13201 CAG0O1 20368972 Ki = 872 nM T13201 C15BEG 20694083 Ki = 92 nM T13201 CKR8T2 20970546 Ki = 82.1 nM T13201 CF28QV 21017876 Ki = 8460 nM T13201 CCJ8Q3 21051266 Ki = 54.1 nM T13201 CH15RE 21051367 Ki = 29.3 nM T13201 CV34MD 21149346 Ki = 103 nM T13201 CJGU80 21240387 Ki = 548.3 nM T13201 C18KAH 21297028 Ki > 10000 nM T13201 CPG6C1 21416985 Ki = 450 nM T13201 COG69P 21449436 Ki = 23 nM T13201 C9J1WT 21497848 Ki > 10000 nM T13201 CC5W7X 21542156 Ki > 10000 nM T13201 CD0K1C 21600238 Ki > 10000 nM T13201 C61KUX 21726402 Ki = 48.1 nM T13201 C54IUM 21778115 Ki = 35120 nM T13201 C27BJH 21778117 Ki = 34410 nM T13201 CJ4O2E 21806575 Ki = 8.7 nM T13201 CO2U7W 21855445 Ki = 3714 nM T13201 CZ45AO 21878638 Ki = 2508.6 nM T13201 C4XAO7 21879009 Ki = 1291.3 nM T13201 CBS63Q 21879398 Ki = 454.3 nM T13201 C02IPY 21978067 Ki = 780 nM T13201 C6IZW0 22132896 Ki > 10000 nM T13201 C9U4TE 22313850 Ki = 24700 nM T13201 CX4Z1D 22315539 Ki = 1789 nM T13201 C81ROV 22316829 Ki = 19081 nM T13201 CPR25C 22706805 Ki = 24400 nM T13201 C09ACH 22833027 Ki = 11 nM T13201 C9W4IA 22836851 Ki = 11 nM T13201 CXR35D 22864792 Ki = 15 nM T13201 CWM8S4 22953340 Ki = 15 nM T13201 C2D8ZL 23111570 Ki = 37 nM T13201 CE8C1R 23228497 Ki = 13 nM T13201 C2DOR4 23263451 Ki > 10000 nM T13201 C9KMP4 23275795 Ki = 48.1 nM T13201 CICR37 23426698 Ki = 61140 nM T13201 CY6D4N 23644659 Ki = 17 nM T13201 C8UIC6 23644662 Ki = 20000 nM T13201 CCLA40 23644663 Ki = 23000 nM T13201 CD5KT2 23644664 Ki = 4200 nM T13201 C1AVT7 23644700 Ki = 290 nM T13201 C52YRI 23645366 Ki = 18 nM T13201 C3BSJ4 23645367 Ki = 10 nM T13201 CE50QI 23645368 Ki = 275 nM T13201 CNL51U 23645369 Ki = 9.5 nM T13201 CPRX73 23645370 Ki = 85 nM T13201 CSZ6J4 23645528 Ki = 121 nM T13201 C6UH9Q 23645529 Ki = 84 nM T13201 CD0JP3 23645530 Ki = 88 nM T13201 CM37EC 23645531 Ki = 140 nM T13201 C9PD5F 23645532 Ki > 200 nM T13201 C1OE7R 23645533 Ki > 200 nM T13201 CCSN04 23645534 Ki > 200 nM T13201 CU08WI 23645535 Ki > 200 nM T13201 CY41UC 23645536 Ki > 200 nM T13201 CX15EH 23645537 Ki > 200 nM T13201 CD3Q6G 23645538 Ki > 200 nM T13201 CE6NQ2 23645539 Ki = 1800 nM T13201 C4VK3U 23645540 Ki = 1600 nM T13201 C8VM1C 23645541 Ki = 19000 nM T13201 C0MUT6 23645542 Ki = 57000 nM T13201 CNI07H 23645543 Ki = 17000 nM T13201 CHK2X1 23645544 Ki = 15000 nM T13201 CW1V2Z 23645545 Ki = 17000 nM T13201 C6SP7T 23645546 Ki = 41000 nM T13201 CD9QO2 23645547 Ki = 30000 nM T13201 C25YLZ 23645548 Ki = 25000 nM T13201 C9WT2E 23645682 Ki = 3400 nM T13201 CU1OK9 23645683 Ki = 3300 nM T13201 CLHE50 23645684 Ki = 14000 nM T13201 C0UXY9 23646323 Ki = 2400 nM T13201 C3QLX1 23646324 Ki = 2700 nM T13201 CMX1A6 23646325 Ki = 4900 nM T13201 C29HMI 23646326 Ki = 7.7 nM T13201 CCW81X 23647027 Ki = 5800 nM T13201 CE20BX 23647028 Ki = 8.5 nM T13201 CNS87E 23661710 Ki = 2550 nM T13201 C8YRU5 23661711 Ki = 8640 nM T13201 CPGY29 23662344 Ki = 8790 nM T13201 C1T3BP 23663627 Ki = 9060 nM T13201 CRZT32 23665339 Ki = 252 nM T13201 C7V6YP 23665706 Ki > 10000 nM T13201 CH5BD7 23665763 Ki = 18000000 nM T13201 CXWP91 23666732 Ki = 0.97 nM T13201 C6W2BA 23668541 Ki = 531 nM T13201 CU08IW 23670409 Ki > 2000 nM T13201 C1HCX5 23671974 Ki = 48 nM T13201 C6F9NR 23672331 Ki = 450000 nM T13201 C21XEP 23672490 Ki = 98000 nM T13201 CYO7C3 23673162 Ki = 310000 nM T13201 CZNV20 23673832 Ki = 300000 nM T13201 CDB01O 23674157 Ki = 909 nM T13201 C4UFA0 23674499 Ki = 120000 nM T13201 CPI26E 23677888 Ki = 3880 nM T13201 CR7O3Q 23677931 Ki = 9.2 nM T13201 CKL59B 23679442 Ki = 76.1 nM T13201 CNIF07 23681162 Ki = 4040 nM T13201 CJA07G 23685506 Ki = 6920 nM T13201 CC93FA 23686905 Ki = 4.1 nM T13201 CZD6O0 23688497 Ki = 795 nM T13201 C54XWY 23689557 Ki = 3880 nM T13201 CH0QD2 23690451 Ki = 7390 nM T13201 C45EHX 23690537 Ki = 101000 nM T13201 C7LE5M 23690998 Ki = 8000 nM T13201 CE52UX 23691027 Ki = 7610 nM T13201 CE91KL 23691977 Ki = 638 nM T13201 CBU67Z 23691979 Ki = 8180 nM T13201 CE03MX 23692005 Ki = 92000 nM T13201 CK2Q0I 23697126 Ki = 425 nM T13201 C4XE6Y 23699059 Ki = 3940 nM T13201 CR41LS 23703293 Ki = 380000 nM T13201 CPX0I4 24204718 Ki = 397 nM T13201 CF83JT 24204719 Ki = 302 nM T13201 CSWR58 24204720 Ki = 405 nM T13201 CIQ9L6 24204924 Ki = 455 nM T13201 CL2V5T 24204925 Ki = 433 nM T13201 C14RLU 24204932 Ki = 336 nM T13201 CN5ST6 24206002 Ki = 498 nM T13201 CPD4Z6 24206003 Ki = 593 nM T13201 C1Y2JB 24286289 Ki = 68.2 nM T13201 CKE1A3 24416843 Ki = 47.3 nM T13201 CA3Y8I 24588559 Ki = 549 nM T13201 CG98KI 24588612 Ki = 752 nM T13201 CK79DN 24588735 Ki = 381 nM T13201 CGHW54 24640576 Ki = 1892.3 nM T13201 C01LHS 24640776 Ki = 85 nM T13201 CT8O2Z 24643222 Ki = 91.1 nM T13201 CB6WE3 24650532 Ki = 847 nM T13201 C1I9HZ 24692821 Ki = 78.4 nM T13201 C8BL9O 24762836 Ki = 5480 nM T13201 CQG9O0 24816432 Ki = 15 nM T13201 CX10RQ 24823136 Ki = 2500 nM T13201 CAS51H 24823137 Ki = 48 nM T13201 CXV0A1 24823299 Ki = 1.6 nM T13201 CK0D4U 24823300 Ki = 9.4 nM T13201 CU6VO3 24823301 Ki = 4400 nM T13201 C8A9PE 24823302 Ki = 4300 nM T13201 C5W7AC 24823303 Ki = 4400 nM T13201 CZMT56 24823304 Ki = 4300 nM T13201 CB9U5Z 24823476 Ki = 5000 nM T13201 CXT1C5 24823477 Ki = 5300 nM T13201 CBDO71 24823478 Ki = 10.5 nM T13201 CUT3V8 24823479 Ki = 9.3 nM T13201 C3UYV0 24823480 Ki = 5000 nM T13201 CJQ3M4 24823631 Ki = 560 nM T13201 CPQN52 24823632 Ki = 2.8 nM T13201 CN75LK 24823633 Ki = 2.5 nM T13201 CV5YR0 24843241 Ki = 260 nM T13201 CNR3U7 24866945 IC50 > 10000 nM T13201 CQRZ10 24877657 Ki = 87 nM T13201 C15OJW 24966977 Ki = 654 nM T13201 C2JQ7M 25040103 Ki = 586 nM T13201 C62DIS 25048179 Ki = 7214 nM T13201 CTVO94 25071013 Ki = 3000 nM T13201 CB0E2M 25071014 Ki = 2200 nM T13201 COI25U 25131351 Ki = 189 nM T13201 CNMY17 25131685 Ki = 242 nM T13201 CB7V8Y 25147773 Ki = 730 nM T13201 CG0S7T 25154732 Ki = 102 nM T13201 CYG1H9 25154741 Ki = 5850 nM T13201 C3KF1V 25178145 Ki = 95 nM T13201 C8PMK7 25178356 Ki = 2339 nM T13201 C9HZG2 25181078 Ki = 116 nM T13201 CMYP34 25181079 Ki = 3430 nM T13201 C7U1YC 25181080 Ki = 1765 nM T13201 C85HLG 25181081 Ki = 2487 nM T13201 C4M9XV 25242508 Ki = 354000 nM T13201 CU14KG 25258358 Ki = 88700 nM T13201 CQ1WE2 25258360 Ki > 200000 nM T13201 CL5EZ6 25258361 Ki = 62200 nM T13201 COU19V 25258363 Ki > 200000 nM T13201 C5T1NZ 25294048 Ki = 4812.1 nM T13201 CRP6F5 25335375 Ki = 8.6 nM T13201 CPN2T5 25392418 Ki = 626.4 nM T13201 C1AOB3 25981084 Ki = 635.9 nM T13201 CP02LF 26365005 Ki = 101 nM T13201 C0RF4D 26470767 Ki > 100000 nM T13201 CMUT78 26500397 Ki = 630.3 nM T13201 C5EC2T 26535209 Ki = 6.8 nM T13201 CLNR46 26598995 Ki > 10000 nM T13201 CA9UZ7 26773685 Ki = 7.7 nM T13201 C8KQ5N 27868059 Ki = 604 nM T13201 CQSA29 27868075 Ki = 6530 nM T13201 C7QB8M 27868953 Ki = 509 nM T13201 CWU2R0 27869227 Ki = 150 nM T13201 C46OQT 27869236 Ki = 49.8 nM T13201 C85HLF 27869237 Ki = 812 nM T13201 C5OWP7 27869350 Ki = 83 nM T13201 CF02EA 27869546 Ki = 76.9 nM T13201 C1G3XO 27869982 Ki = 1465 nM T13201 C8ML3W 27870055 Ki = 5500 nM T13201 CMK25I 27870443 Ki = 470 nM T13201 CQK4O6 27870796 Ki = 388 nM T13201 C2Z4FP 27870803 Ki = 3690 nM T13201 C61AIY 28452155 Ki = 29 nM T13201 C3RG8K 28846439 Ki = 421 nM T13201 C4EB0J 29034199 Ki = 30.7 nM T13201 C0CJ5I 29045530 Ki = 23.5 nM T13201 CF8SA7 29559803 Ki = 20.9 nM T13201 C4R0ZU 29981063 Ki > 10000 nM T13201 CBPO08 34751720 Ki = 7966.7 nM T13201 CVXO26 35053285 Ki = 38 nM T13201 CF3HA1 35871284 Ki = 430 nM T13201 CI0K1J 36865965 Ki = 9.2 nM T13201 C5IUO9 38154971 Ki = 3260 nM T13201 CZE95V 38155699 Ki = 1680 nM T13201 CSB4C7 38159448 Ki = 4800 nM T13201 C4F7YT 40086402 Ki = 1342 nM T13201 C06EUO 40662472 Ki = 189 nM T13201 C1U4TL 41180562 Ki = 73 nM T13201 CH2P6W 41430216 Ki = 5530 nM T13201 C5YBO2 41484755 Ki = 1700 nM T13201 CUK13R 41874556 Ki > 10000 nM T13201 C0J8DM 42597612 Ki = 4340 nM T13201 C8A5CF 42597613 Ki = 3710 nM T13201 C58ZUN 42597614 Ki = 3970 nM T13201 COG2A0 42597615 Ki = 4680 nM T13201 C1J9CQ 42597616 Ki = 3710 nM T13201 COG2I5 42598921 Ki = 4120 nM T13201 CDXS12 42598922 Ki = 4150 nM T13201 C6WU8M 42609905 Ki = 3.5 nM T13201 CP7UM8 42643988 Ki = 290000 nM T13201 C0IE3B 42644449 Ki = 548000 nM T13201 CT2C3D 42644450 Ki = 508000 nM T13201 CYJ0H4 43089860 Ki = 187 nM T13201 CNB1E8 43139163 Ki = 189.5 nM T13201 CXJY80 43235186 Ki = 4.4 nM T13201 CC5TY6 43321518 Ki = 228.3 nM T13201 C23CNV 43321585 Ki = 209.5 nM T13201 C7EO2A 43329592 Ki = 246 nM T13201 CA0DX4 43342474 Ki = 315 nM T13201 C2HY4R 43342475 Ki = 207 nM T13201 CBK0M6 43342481 Ki = 143 nM T13201 C41VHR 43468983 Ki = 94.9 nM T13201 C82MRL 44144383 Ki = 50.9 nM T13201 CUT9E0 44186130 Ki = 6.5 nM T13201 C8D7UR 44186132 Ki = 7.6 nM T13201 CL08CN 44186134 Ki = 35.3 nM T13201 C3UC8S 44186136 Ki = 31.8 nM T13201 CXT6O8 44186138 Ki = 25.1 nM T13201 CLP2V8 44186201 Ki = 5.2 nM T13201 CEN2Y5 44186203 Ki = 1.5 nM T13201 CYR23T 44186205 Ki = 0.92 nM T13201 CAF52T 44186207 Ki = 0.93 nM T13201 CZR5W4 44186209 Ki = 9.3 nM T13201 C4POV2 44186263 Ki = 9.7 nM T13201 CW95CB 44186265 Ki = 20.9 nM T13201 CQ6JB5 44186267 Ki = 3.2 nM T13201 C1REF8 44186269 Ki = 0.98 nM T13201 CZM6N5 44186271 Ki = 0.97 nM T13201 CCXN08 44219644 Ki = 2900 nM T13201 C82GHC 44219651 Ki = 2700 nM T13201 CW1Q9E 44219652 IC50 = 158 nM T13201 C49UTC 44219653 IC50 = 520 nM T13201 C36OBU 44219661 IC50 = 120 nM T13201 CI2LS6 44221745 Ki = 39 nM T13201 CAY8B9 44221746 Ki = 39 nM T13201 CP1K7W 44221747 Ki > 100000 nM T13201 CFEJ21 44221748 Ki = 8960 nM T13201 CZ9X2W 44221749 Ki = 65 nM T13201 C8T4IC 44221941 Ki = 3490 nM T13201 CJE2D7 44221942 Ki = 620 nM T13201 CERA26 44221943 Ki = 35 nM T13201 C7TJF2 44221944 Ki > 100000 nM T13201 CG2D4X 44268930 Ki = 105 nM T13201 CX1CK5 44268931 Ki = 200 nM T13201 CZT39W 44268932 Ki = 2400 nM T13201 C6ECO2 44268933 Ki = 760 nM T13201 C15VUL 44268934 Ki = 240 nM T13201 CO83EW 44269005 Ki = 2 nM T13201 C8T3FR 44269010 Ki = 5 nM T13201 C9LUN8 44269014 Ki = 11500 nM T13201 C5HTZ4 44269015 Ki = 950 nM T13201 CE07DX 44269023 Ki > 50000 nM T13201 CD71PZ 44269025 Ki = 800 nM T13201 CM1SO2 44269027 Ki = 630 nM T13201 CIZ2H8 44269028 Ki = 10000 nM T13201 C53OWA 44269034 Ki = 24000 nM T13201 C0Y8PD 44269040 Ki = 31 nM T13201 CJ4CQ2 44269056 Ki = 560 nM T13201 CHQT54 44269066 Ki = 15000 nM T13201 CARG97 44269072 Ki = 500 nM T13201 CB59ZH 44269073 Ki = 3000 nM T13201 CZ5G4I 44295070 Ki = 205 nM T13201 CZH4J1 44295071 Ki = 210 nM T13201 C4TKI3 44295073 Ki = 38 nM T13201 C5N9HB 44295232 Ki = 30 nM T13201 C5SJ8L 44295325 Ki = 435 nM T13201 C8V4GI 44295335 Ki = 130 nM T13201 C63FNX 44295336 Ki = 175 nM T13201 CFQ3Z0 44295339 Ki = 415 nM T13201 CNR6G2 44295340 Ki = 425 nM T13201 CM1V4E 44295349 Ki = 200 nM T13201 C9G5AI 44295381 Ki = 405 nM T13201 C7R6JT 44295382 Ki = 250 nM T13201 CWFN72 44295388 Ki = 15 nM T13201 C1K8SN 44295397 Ki = 54 nM T13201 CM7AJ8 44295411 Ki = 39 nM T13201 CYBT62 44295448 Ki = 36 nM T13201 C20PFZ 44295453 Ki = 41 nM T13201 C13NTV 44295458 Ki = 69 nM T13201 CUIB83 44295459 Ki = 100 nM T13201 C0AGJ6 44295464 Ki = 27 nM T13201 C2N6AL 44295477 Ki = 135 nM T13201 C1RVC6 44295493 Ki = 115 nM T13201 CGAJ68 44295497 Ki = 103 nM T13201 CF8Q3E 44295519 Ki = 380 nM T13201 C38CMP 44295539 Ki = 270 nM T13201 C9K8WR 44295565 Ki = 250 nM T13201 CE49OS 44295574 Ki = 300 nM T13201 CV1LQ8 44295581 Ki = 425 nM T13201 CEV72P 44295589 Ki = 285 nM T13201 C7C5BP 44295596 Ki = 320 nM T13201 C18IXK 44295597 Ki = 170 nM T13201 C6WG1X 44295602 Ki = 240 nM T13201 CU4O3K 44295612 Ki = 37 nM T13201 C6J3EG 44295620 Ki = 440 nM T13201 CAQ28E 44295627 Ki = 150 nM T13201 C90FBC 44295647 Ki = 125 nM T13201 CB2J7Q 44295734 Ki = 40 nM T13201 C8B1EU 44295749 Ki = 400 nM T13201 CAQ8D5 44295756 Ki = 35 nM T13201 C5Z7KR 44295772 Ki = 320 nM T13201 C8SE3Z 44295795 Ki = 535 nM T13201 CCI7X0 44295824 Ki = 305 nM T13201 C8MVP1 44295825 Ki = 240 nM T13201 C4M1WH 44295835 Ki = 240 nM T13201 CYM91I 44295843 Ki = 520 nM T13201 CJ0S8N 44295871 Ki = 425 nM T13201 CH36RU 44295906 Ki = 420 nM T13201 CWY05P 44295942 Ki = 450 nM T13201 CFZN67 44295943 Ki = 475 nM T13201 CC68PJ 44295959 Ki = 400 nM T13201 CG14BN 44295994 Ki = 430 nM T13201 CGCE21 44296010 Ki = 410 nM T13201 C1VKH3 44296089 Ki = 560 nM T13201 COGP36 44296104 Ki = 270 nM T13201 C6V9WT 44309709 Ki = 278 nM T13201 CYUE74 44309710 Ki = 31 nM T13201 CERI42 44309802 Ki = 33 nM T13201 CLBU37 44310092 Ki = 315 nM T13201 CW0S8U 44311169 Ki = 31 nM T13201 C0B4HZ 44312333 Ki > 200 nM T13201 C76HLZ 44314854 Ki = 3 nM T13201 C91HDR 44315566 Ki > 10000 nM T13201 C4T7BJ 44322528 Ki = 15 nM T13201 CV72ZF 44322583 Ki = 2000 nM T13201 CG0RI3 44322584 Ki = 2050 nM T13201 CXDA80 44322970 Ki = 16 nM T13201 CLQS83 44327323 Ki = 210 nM T13201 CPTU85 44329131 Ki = 16 nM T13201 C7X5HT 44329132 Ki = 20 nM T13201 CK2O4V 44329147 Ki = 16 nM T13201 CEU58D 44329411 Ki = 12 nM T13201 CNLO86 44329422 Ki = 45 nM T13201 CI6AW0 44329423 Ki = 12 nM T13201 C6DKW1 44329437 Ki = 15 nM T13201 C3RFO4 44329445 Ki = 13 nM T13201 CI9KS2 44329453 Ki = 12 nM T13201 CU78BY 44329463 Ki = 15 nM T13201 CX2HZ1 44329466 Ki = 13 nM T13201 CR13HU 44329471 Ki = 14 nM T13201 C7U0QG 44329472 Ki = 14 nM T13201 COZ8Q4 44329485 Ki = 68 nM T13201 CC85EH 44329560 Ki = 13 nM T13201 CNY0R6 44329561 Ki = 11 nM T13201 CX0W5V 44329576 Ki = 73 nM T13201 C6BGE3 44329679 Ki = 17 nM T13201 CP67GZ 44329699 Ki = 13 nM T13201 CM21EZ 44329700 Ki = 15 nM T13201 CQY2H4 44329734 Ki = 15 nM T13201 CPG0U9 44329736 Ki = 16 nM T13201 C4D9HU 44329737 Ki = 50 nM T13201 CU41NJ 44329768 Ki = 17 nM T13201 CS7D6E 44329771 Ki = 23 nM T13201 CBK4M3 44329804 Ki = 18 nM T13201 C7G4IN 44329805 Ki = 16 nM T13201 CH43UT 44332605 Ki = 15 nM T13201 CWRD02 44332665 Ki = 13 nM T13201 CP0WO3 44338600 Ki = 5.5 nM T13201 CFJD87 44345920 Ki = 80 nM T13201 C3XJK5 44346012 Ki = 50 nM T13201 CKI8S2 44347455 Ki = 1700 nM T13201 C3T5BJ 44347553 Ki = 9 nM T13201 CK62UO 44347554 Ki = 12 nM T13201 CFHX13 44347728 Ki = 1800 nM T13201 C8MJ2U 44347729 Ki = 9 nM T13201 CKA91T 44347760 Ki = 1500 nM T13201 CCJ82U 44347774 Ki = 1500 nM T13201 C0ZAW1 44347825 Ki = 11 nM T13201 C4O3KI 44347826 Ki = 1000 nM T13201 CUT7R6 44347834 Ki = 1200 nM T13201 C18YIR 44347836 Ki = 9 nM T13201 CL53AZ 44347837 Ki = 11 nM T13201 C0AXH3 44347849 Ki = 78 nM T13201 CLXC41 44347889 Ki = 1300 nM T13201 CR0X1H 44347896 Ki = 10 nM T13201 C3WA6I 44347907 Ki = 16 nM T13201 CRU7E6 44347909 Ki = 11 nM T13201 C0VS9L 44347924 Ki = 1500 nM T13201 C4T6SW 44359832 Ki = 250 nM T13201 CL6WK9 44359987 Ki = 350 nM T13201 CXBM69 44360292 Ki = 380 nM T13201 CQ3G7E 44363244 Ki = 25 nM T13201 C83HZB 44363263 Ki = 30 nM T13201 C5NGZ6 44363316 Ki = 115 nM T13201 C6T7KR 44363320 Ki = 110 nM T13201 CXG27B 44363365 Ki = 28 nM T13201 CL8QM1 44363386 Ki = 97 nM T13201 C8GC9V 44363414 Ki = 54 nM T13201 CB2JK5 44363440 Ki = 26 nM T13201 C6ETL2 44363444 Ki = 20 nM T13201 CT8QU4 44363445 Ki = 35 nM T13201 C0DTE3 44363462 Ki = 50 nM T13201 CITL93 44363515 Ki = 40 nM T13201 C5I2YQ 44363519 Ki = 38 nM T13201 CH4YN1 44363520 Ki = 27 nM T13201 CM6O2J 44363524 Ki = 23 nM T13201 C9S6NA 44363540 Ki = 27 nM T13201 COQM57 44363589 Ki = 23 nM T13201 C10PKB 44363655 Ki = 23 nM T13201 CL8OU3 44363657 Ki = 21 nM T13201 CYE04Z 44363692 Ki = 13 nM T13201 C1IM4R 44363714 Ki = 35 nM T13201 CA40KV 44363764 Ki = 22 nM T13201 CDN4K1 44363803 Ki = 21 nM T13201 CAPN36 44367390 Ki = 38000 nM T13201 CS4P3F 44367405 Ki = 100 nM T13201 CD98KU 44367410 Ki = 410 nM T13201 CF8J7B 44367431 Ki = 400 nM T13201 CE18VJ 44367432 Ki > 1000000 nM T13201 CT0R9B 44367463 Ki = 430 nM T13201 CHE0B6 44373668 Ki = 21800 nM T13201 CLQK83 44373669 Ki = 540 nM T13201 CZ01KF 44373682 Ki = 20000 nM T13201 CLA0S6 44373694 Ki = 1060 nM T13201 CY9NC0 44373699 Ki = 600 nM T13201 C1NT8P 44373700 Ki = 520 nM T13201 C8LSM2 44373716 Ki = 18000 nM T13201 CGRJ30 44373728 Ki = 610 nM T13201 C0T5BN 44373729 Ki = 36 nM T13201 CJ4HY3 44373738 Ki = 33 nM T13201 CCQ89X 44373741 Ki = 1 nM T13201 CI34UE 44373906 Ki = 21500 nM T13201 C4B7LG 44373919 Ki = 15000 nM T13201 C63UGJ 44373942 Ki = 950 nM T13201 CPG1U2 44373981 Ki = 39 nM T13201 C3SQF9 44373982 Ki = 400 nM T13201 CH8F9D 44373983 Ki = 500 nM T13201 CIX89D 44380403 Ki > 100000 nM T13201 CR8UH5 44380428 Ki = 420000 nM T13201 CZHX52 44380431 Ki = 1200 nM T13201 CJVY96 44380588 Ki = 18 nM T13201 CCLG64 44380603 Ki = 149 nM T13201 CBC73O 44380656 Ki > 100000 nM T13201 C4M7PV 44380677 Ki > 100000 nM T13201 CT3CM0 44380678 Ki > 100000 nM T13201 CM0V9I 44380939 Ki = 39 nM T13201 CXY9F6 44380940 Ki = 62 nM T13201 C3XN9Y 44380951 Ki = 17 nM T13201 CUV2W6 44380955 Ki = 26 nM T13201 CKT4J7 44381089 Ki = 750 nM T13201 C1M4GF 44381090 Ki = 400000 nM T13201 C6K9PD 44381123 Ki > 100000 nM T13201 CVB7U8 44381140 Ki = 960 nM T13201 C5O9LH 44389667 Ki = 95 nM T13201 CL5GF2 44389703 Ki = 77 nM T13201 C9DRN1 44389734 Ki = 113 nM T13201 CE9BS6 44389758 Ki = 54 nM T13201 C68TCP 44389772 Ki = 61 nM T13201 C9OM5F 44389791 Ki = 63 nM T13201 C7VMQ6 44389836 Ki = 80 nM T13201 CF19RI 44389844 Ki = 250 nM T13201 CG2U5A 44389881 Ki = 73 nM T13201 CR16DV 44389954 Ki = 135 nM T13201 C8KE4X 44389960 Ki = 24 nM T13201 CEV89Z 44389961 Ki = 50 nM T13201 C5ZCF3 44389968 Ki = 72 nM T13201 C06AUB 44389978 Ki = 40 nM T13201 C09EFT 44389990 Ki = 24 nM T13201 CFBU06 44389993 Ki = 79 nM T13201 C3IBQ1 44389995 Ki = 74 nM T13201 CP8JK3 44390019 Ki = 54 nM T13201 CWCQ49 44390027 Ki = 324 nM T13201 CVW6E1 44390031 Ki = 33 nM T13201 C5TO9D 44390032 Ki = 313 nM T13201 CI8PB1 44391626 Ki = 93 nM T13201 C68BRH 44391633 Ki = 267 nM T13201 C6BUC8 44391791 Ki = 7.9 nM T13201 CWR3F1 44391802 Ki = 644 nM T13201 CM6F7X 44391805 Ki = 8.2 nM T13201 C93OPV 44391820 Ki = 7.6 nM T13201 CDH40E 44391824 Ki = 9.6 nM T13201 CUK9X4 44391833 Ki = 7.1 nM T13201 COTH27 44391859 Ki = 820 nM T13201 CD9H6W 44392389 Ki = 31 nM T13201 C5ZA9R 44395106 Ki = 88 nM T13201 C4OR5F 44395107 Ki = 85 nM T13201 C9J2ME 44395133 Ki = 75 nM T13201 C9MLB4 44395134 Ki = 103 nM T13201 CI3O9B 44395149 Ki = 83 nM T13201 CO8J7I 44395150 Ki = 90 nM T13201 CPB8W7 44395163 Ki = 136 nM T13201 C8EK1N 44395173 Ki = 94 nM T13201 CQ54DL 44395174 Ki = 96 nM T13201 CWUP51 44395202 Ki = 78 nM T13201 CIWO28 44395243 Ki = 116 nM T13201 CYR62U 44395244 Ki = 105 nM T13201 CUW0D8 44395258 Ki = 82 nM T13201 C6H1QR 44395691 Ki = 0.6 nM T13201 CWN75T 44395718 Ki = 0.7 nM T13201 CR81IG 44395747 Ki = 0.7 nM T13201 CYS09N 44395778 Ki = 15 nM T13201 CMSJ40 44395790 Ki = 7.2 nM T13201 CD4AX9 44395811 Ki = 1.6 nM T13201 CX9RC2 44395866 Ki = 0.6 nM T13201 CN7A1U 44395892 Ki = 24 nM T13201 C90XMR 44395897 Ki = 58 nM T13201 CVC7K9 44395919 Ki = 60 nM T13201 CL5FR8 44396970 Ki = 53 nM T13201 CY4L9G 44396983 Ki = 64 nM T13201 C3CB6J 44397074 Ki = 31 nM T13201 CWBC15 44397108 Ki = 58 nM T13201 C3VG4H 44397112 Ki = 197 nM T13201 C65XZL 44397209 Ki = 25 nM T13201 CFK1W2 44397213 Ki = 31 nM T13201 CX1V2T 44397238 Ki = 23 nM T13201 C6Y5MJ 44397294 Ki = 42 nM T13201 C5Z7FC 44397318 Ki = 29 nM T13201 CA65VH 44398374 Ki = 7000 nM T13201 C7T8XG 44399285 Ki = 247 nM T13201 CNSR28 44399286 Ki = 156 nM T13201 C8NOW9 44399298 Ki = 105 nM T13201 C89LNG 44399317 Ki = 93 nM T13201 CT3V7P 44399318 Ki = 3500 nM T13201 CCD34Q 44399321 Ki = 76 nM T13201 C67HFO 44399335 Ki = 368 nM T13201 CQJZ93 44399338 Ki = 70 nM T13201 C0KFU7 44399339 Ki = 49 nM T13201 CH6GT7 44399340 Ki = 34 nM T13201 CG0Z9A 44399346 Ki = 622 nM T13201 C8EQG2 44399347 Ki = 549 nM T13201 C5GJ3N 44399351 Ki = 39 nM T13201 CNTM52 44399371 Ki = 235 nM T13201 C3QZR6 44399393 Ki = 130 nM T13201 C7BHR6 44399404 Ki = 113 nM T13201 C7LCX4 44399427 Ki = 180 nM T13201 C48MQR 44399437 Ki = 561 nM T13201 CCZG27 44399440 Ki = 95 nM T13201 C72HQK 44399449 Ki = 91 nM T13201 CGEX61 44399456 Ki = 631 nM T13201 CU1B9T 44399459 Ki = 558 nM T13201 CV9EU2 44399460 Ki = 1560 nM T13201 CQCB53 44399461 Ki = 1635 nM T13201 CZ4DF9 44399462 Ki = 33 nM T13201 CZ3YC5 44399486 Ki = 112 nM T13201 CVK1X8 44399489 Ki = 241 nM T13201 CUK37Q 44399499 Ki = 128 nM T13201 CVP43X 44399501 Ki = 176 nM T13201 CRM73I 44399515 Ki = 104 nM T13201 CK6G2Y 44399516 Ki = 4200 nM T13201 C4UEG1 44399517 Ki = 8500 nM T13201 CL6F3X 44399532 Ki = 540 nM T13201 CU7BK9 44399535 Ki = 31 nM T13201 CX6B8J 44399541 Ki = 425 nM T13201 CMFY95 44399542 Ki = 198 nM T13201 C8B9NK 44399547 Ki = 875 nM T13201 CT57KL 44399549 Ki = 87 nM T13201 CB0R2P 44399570 Ki = 613 nM T13201 CD5MJ6 44399571 Ki = 35 nM T13201 C3EBD7 44399585 Ki = 69 nM T13201 C0RT3E 44399598 Ki = 69 nM T13201 CPKG57 44399624 Ki = 36 nM T13201 CI5Y0H 44399639 Ki = 70.5 nM T13201 C2T7MB 44399654 Ki = 92 nM T13201 CU3DY1 44399655 Ki = 94 nM T13201 C4AD1R 44399664 Ki = 70 nM T13201 CR95YM 44399687 Ki = 72 nM T13201 CGC2M5 44399695 Ki = 70 nM T13201 C3W9CF 44399734 Ki = 77 nM T13201 CUXT35 44401673 Ki = 210 nM T13201 C4AD6B 44401689 Ki = 9.5 nM T13201 C1A5NV 44401728 Ki = 246 nM T13201 CWJ08B 44401743 Ki = 7300 nM T13201 C9O1UL 44401744 Ki = 8200 nM T13201 C27YCF 44401745 Ki = 8100 nM T13201 C83EIL 44401769 Ki = 233 nM T13201 C2HDZ6 44401810 Ki = 9000 nM T13201 CJ86PU 44401826 Ki = 105 nM T13201 C0F1VY 44401832 Ki = 8600 nM T13201 CQ02ZD 44401833 Ki = 4000 nM T13201 C5PR9E 44401857 Ki = 3.1 nM T13201 C7NM9T 44401871 Ki = 8300 nM T13201 CD9I8V 44401873 Ki = 6000 nM T13201 CYQF42 44401889 Ki = 175 nM T13201 CIN38J 44401926 Ki = 254000 nM T13201 C75WFG 44401951 Ki = 303000 nM T13201 CX1LH3 44401952 Ki = 268 nM T13201 CIO61G 44401975 Ki = 308000 nM T13201 C9M0ID 44401978 Ki = 7600 nM T13201 CU53CI 44401994 Ki = 5800 nM T13201 C34PLI 44402062 Ki = 249000 nM T13201 CF6X9Y 44402148 Ki = 308 nM T13201 C28JBO 44402274 Ki = 355 nM T13201 CGPF38 44402275 Ki = 3.7 nM T13201 CT6UF5 44402709 Ki = 29 nM T13201 C5FC0Y 44402716 Ki > 1000 nM T13201 C8N0GW 44402748 Ki = 44 nM T13201 C9AJ7Z 44402772 Ki = 35 nM T13201 CR72VG 44402825 Ki = 94 nM T13201 C5LU4G 44403258 Ki = 85 nM T13201 C6OS3R 44403265 Ki = 290 nM T13201 CI18FK 44403266 Ki = 530 nM T13201 CR2Z7F 44403267 Ki = 493 nM T13201 C0W6BQ 44403268 Ki > 1000 nM T13201 C8QXA6 44403278 Ki > 1000 nM T13201 CSN79Y 44403312 Ki = 245 nM T13201 CW93DL 44405187 Ki = 98 nM T13201 CSXF07 44405190 Ki = 415 nM T13201 CQN4P8 44408881 Ki = 12150 nM T13201 COM50H 44408887 Ki = 12045 nM T13201 CVJ5T9 44416166 Ki = 19700 nM T13201 CZT1U9 44416167 Ki = 7800 nM T13201 CQ36IP 44416168 Ki = 6400 nM T13201 CS49FE 44416185 Ki = 11600 nM T13201 CEH5P1 44416186 Ki = 27300 nM T13201 C8C4IJ 44416203 Ki = 220000 nM T13201 CE6N7Q 44416215 Ki = 113000 nM T13201 CY9VT1 44416239 Ki = 7300 nM T13201 CI01QM 44416240 Ki = 10900 nM T13201 CX8ZQ9 44416241 Ki = 392000 nM T13201 CRX27F 44416256 Ki = 310000 nM T13201 C68YLB 44416306 Ki = 5800 nM T13201 C5ROE2 44416307 Ki = 7700 nM T13201 C47OTU 44416317 Ki = 14200 nM T13201 CE4M9P 44416378 Ki = 22100 nM T13201 CE03DL 44416379 Ki = 82100 nM T13201 C67IEM 44420782 Ki = 5200 nM T13201 CY49HT 44423674 Ki = 8910 nM T13201 CHI5G1 44423675 Ki = 880 nM T13201 CFC3M6 44423676 Ki = 156000 nM T13201 CO24JF 44423677 Ki = 4100 nM T13201 C7F9DB 44423678 Ki = 890 nM T13201 CJ6GW5 44423679 Ki = 900 nM T13201 CUKM29 44423680 Ki = 5900 nM T13201 C3R0FS 44423681 Ki = 9000 nM T13201 C14DBJ 44423682 Ki = 9700 nM T13201 CA90GQ 44424362 Ki > 200000 nM T13201 C5HB4P 44424363 Ki = 9350 nM T13201 CK8S7Y 44424364 Ki > 200000 nM T13201 C28QYE 44424366 Ki = 6880 nM T13201 CP3OY8 44428369 Ki = 583 nM T13201 CM3J0U 44430517 Ki = 10700 nM T13201 C9LT7Y 44430518 Ki = 11000 nM T13201 C1VTB6 44430520 Ki = 10200 nM T13201 C2L5MB 44430521 Ki = 12300 nM T13201 CVEO17 44430523 Ki = 13300 nM T13201 C8MFL1 44430524 Ki = 9400 nM T13201 CW8DJ9 44435841 Ki = 7100 nM T13201 CQ4RC2 44435843 Ki = 3000 nM T13201 C9RYT1 44435845 Ki = 8540 nM T13201 CHDA78 44435846 Ki = 26160 nM T13201 C1G7HL 44435848 Ki = 3280 nM T13201 CW3M0X 44435849 Ki = 18740 nM T13201 CA4ZH8 44435850 Ki = 71620 nM T13201 CW73VG 44435851 Ki = 30770 nM T13201 C3D6AL 44435853 Ki = 222820 nM T13201 C6X5NI 44435855 Ki = 7110 nM T13201 COUY42 44435856 Ki = 125000 nM T13201 C1LM4Y 44435857 Ki = 9090 nM T13201 CU72AI 44435858 Ki = 4320 nM T13201 C5AMH4 44435861 Ki = 4310 nM T13201 C38GXC 44435862 Ki = 144070 nM T13201 C1AOX2 44435863 Ki = 42250 nM T13201 CFBT23 44435864 Ki = 8620 nM T13201 C37DRO 44435865 Ki = 4340 nM T13201 CT3S5B 44435866 Ki = 73250 nM T13201 C3PTQ7 44435867 Ki = 8530 nM T13201 CUO81X 44445087 Ki = 4 nM T13201 CE61WS 44445088 Ki = 4 nM T13201 COS30Z 44445089 Ki = 40 nM T13201 CWGV59 44445090 Ki = 60 nM T13201 CGP58E 44445091 Ki = 200 nM T13201 C72RWK 44445092 Ki = 200 nM T13201 CV4WU5 44445094 Ki = 180 nM T13201 C74ECN 44448778 Ki = 204 nM T13201 CX50NI 44448882 Ki = 179 nM T13201 CNRW48 44448977 Ki = 170 nM T13201 CUWK18 44449006 Ki = 89 nM T13201 CB9KU0 44449032 Ki = 365 nM T13201 CSFE58 44449055 Ki = 784 nM T13201 CV31AN 44449057 Ki = 128 nM T13201 C7PU2N 44449080 Ki = 233 nM T13201 CLIV87 44449082 Ki = 182 nM T13201 C48XSU 44449083 Ki = 2070 nM T13201 C53DYE 44458870 Ki = 950 nM T13201 C7ULS2 44459273 Ki = 250 nM T13201 C23QZG 44459307 Ki = 270 nM T13201 C8P4EB 44459430 Ki = 480 nM T13201 CNW10Y 44459431 Ki = 9.5 nM T13201 CUER27 44511333 IC50 = 7130000 nM T13201 CFW8V2 44520897 Ki = 161 nM T13201 CR4NZ3 44520898 Ki = 77 nM T13201 CI78UO 44520899 Ki = 84 nM T13201 CQUC34 44520900 Ki = 72 nM T13201 CNC1D8 44520905 Ki = 73 nM T13201 CR43NP 44520906 Ki = 63 nM T13201 CHCT21 44542292 Ki = 11 nM T13201 CG61YX 44542293 Ki = 41.5 nM T13201 CL8AQ5 44542294 Ki = 11.1 nM T13201 CF2RX4 44542600 Ki = 9 nM T13201 C5MZ3O 44542742 Ki = 10.1 nM T13201 CI9VZ6 44542743 Ki = 56.5 nM T13201 C8E0MV 44552472 Ki = 3480 nM T13201 CKG53H 44552473 Ki = 2470 nM T13201 C17XAJ 44552559 Ki = 2510 nM T13201 C18XNW 44564181 Ki = 12000 nM T13201 CJ05ZA 44571847 Ki = 6860 nM T13201 C52WIF 44571892 Ki = 103 nM T13201 C64APD 44574189 Ki = 8980 nM T13201 CV5XS1 44574190 Ki = 25700 nM T13201 CE0ZS5 44574217 Ki = 9440 nM T13201 C3OYU7 44574218 Ki = 4070 nM T13201 CHJV65 44574219 Ki = 4430 nM T13201 C4FI0H 44574220 Ki = 3490 nM T13201 CM9E2T 44574221 Ki = 7690 nM T13201 C5MCT7 44574248 Ki = 330 nM T13201 CZB19D 44574249 Ki = 3830 nM T13201 C48VUR 44574250 Ki = 8070 nM T13201 CL96KM 44574828 Ki = 2420 nM T13201 C0AD8M 44574829 IC50 = 210 nM T13201 CGQ1I9 44574914 IC50 = 390 nM T13201 CH03WX 44577410 Ki = 8700 nM T13201 CCH53K 44577411 Ki = 2400 nM T13201 CACY16 44577574 Ki = 6500 nM T13201 CQ3RT6 44577575 Ki = 5800 nM T13201 C03CLH 44577576 Ki = 5500 nM T13201 CKT85S 44577800 Ki = 342 nM T13201 C3DU8S 44577801 Ki = 368 nM T13201 CZ29UX 44577802 Ki = 4000 nM T13201 C5RZK3 44577803 Ki = 100 nM T13201 CB1E6X 44577804 Ki = 4600 nM T13201 CCW3S1 44578981 Ki = 131 nM T13201 CU7Y8T 44578982 Ki = 91 nM T13201 C86YLD 44579460 Ki = 94 nM T13201 CD4WO8 44579535 Ki = 120 nM T13201 CF0KQ8 44581932 Ki = 6 nM T13201 CXD9V3 44590306 Ki > 200000 nM T13201 CM2L4W 44591861 Ki = 60 nM T13201 CSU20V 44591862 Ki = 7 nM T13201 CF9MS6 44591908 Ki = 7 nM T13201 CQ40FB 44592373 Ki = 91 nM T13201 C15THP 44592446 Ki = 103 nM T13201 CDB3X7 44592447 Ki = 97 nM T13201 C2J3ER 44592448 Ki = 117 nM T13201 CUXJ39 44592449 Ki = 80 nM T13201 CTI2C1 44592450 Ki = 79 nM T13201 COS6N0 44592512 Ki = 114 nM T13201 CASL51 44592513 Ki = 102 nM T13201 CXL68J 44592514 Ki = 101 nM T13201 COL03N 44592515 Ki = 60 nM T13201 CHMW14 44592516 Ki = 62 nM T13201 CWG4S1 44629933 Ki = 31700000 nM T13201 CVB2U3 44632018 Ki = 750 nM T13201 COX6D8 45028566 Ki = 89 nM T13201 CF2WL9 45028890 Ki = 1830 nM T13201 C4MO3S 45028891 Ki = 4160 nM T13201 C80CDA 45028892 Ki = 6120 nM T13201 C6YHW4 45028893 Ki = 7130 nM T13201 C16ILW 45028894 Ki = 6100 nM T13201 C5W1RK 45029305 IC50 = 7680 nM T13201 C6T3IO 45029333 IC50 = 8510 nM T13201 CEY71Z 45117541 Ki = 1540 nM T13201 CUQB41 45266944 IC50 = 21000000 nM T13201 C2SHJ7 45266999 Ki > 100000 nM T13201 COE8U0 45267045 Ki > 10000 nM T13201 CM20PR 45267196 Ki = 9500 nM T13201 CA07CZ 45268031 Ki = 6510 nM T13201 C3VB9U 45268767 IC50 = 124000000 nM T13201 C23MVW 45269009 IC50 = 78 nM T13201 C0RG8K 45269749 Ki = 3700 nM T13201 CJX37G 45375967 Ki = 2950 nM T13201 CJ68EO 45375968 Ki = 410 nM T13201 CSE48D 45375973 Ki = 1520 nM T13201 C4LZW6 45483195 Ki = 85 nM T13201 C6E7XJ 45484068 Ki = 4530 nM T13201 CGI25L 45484069 Ki = 3920 nM T13201 CVG6K1 45484072 Ki = 3900 nM T13201 CV5RQ3 45484187 Ki = 78 nM T13201 CTG20B 45485271 Ki = 44700 nM T13201 CK4U0V 45485283 Ki = 145000 nM T13201 CW7FR9 45486144 Ki = 470 nM T13201 C8T4WM 45486167 Ki = 705 nM T13201 C5GZ1B 46197458 Ki = 4160 nM T13201 C3Z7OL 46197569 Ki = 120 nM T13201 CUQF42 46197571 Ki = 6830 nM T13201 C4C7XG 46197572 Ki = 3460 nM T13201 CLBG91 46197677 Ki = 120 nM T13201 C9GC5Q 46197678 Ki = 110 nM T13201 C16XCV 46197680 Ki = 4930 nM T13201 C3JW1R 46197790 Ki = 2040 nM T13201 CD49XQ 46197791 Ki = 102 nM T13201 C4H9TD 46197792 Ki = 87 nM T13201 C0W1GZ 46197794 Ki = 107 nM T13201 CUO20Q 46197893 Ki = 101 nM T13201 CN7KI3 46197894 Ki = 3890 nM T13201 CD74LO 46197895 Ki = 4100 nM T13201 CZ93SW 46197897 Ki = 8040 nM T13201 CNQZ73 46197997 Ki = 6750 nM T13201 CCAX25 46197998 Ki = 90 nM T13201 CQ3R2U 46197999 Ki = 4710 nM T13201 CGM42H 46198111 Ki = 3460 nM T13201 C0DKY8 46198112 Ki = 5570 nM T13201 CBWN61 46198113 Ki = 88 nM T13201 C0AF1L 46198114 Ki = 82 nM T13201 C1KWB5 46198220 Ki = 78 nM T13201 CEV26X 46198221 Ki = 102 nM T13201 CHE08Y 46225608 Ki = 13270 nM T13201 CIE2H3 46225609 Ki = 16320 nM T13201 CF42NR 46225631 Ki = 13830 nM T13201 C0ZG3L 46225639 Ki = 14280 nM T13201 CGW1I5 46225644 Ki = 13260 nM T13201 CEOQ06 46225645 Ki = 2141 nM T13201 CR0WO3 46225646 Ki = 3260 nM T13201 CC2BL5 46225656 Ki = 3290 nM T13201 CW52PZ 46225672 Ki = 2590 nM T13201 CXJ1C9 46225673 Ki = 2460 nM T13201 C6ION5 46236927 Ki = 3590 nM T13201 C7SFG3 46236928 Ki = 2440 nM T13201 CC82QE 46237039 Ki = 3050 nM T13201 CBCK34 46237040 Ki = 1560 nM T13201 CSD29O 46237041 Ki = 1850 nM T13201 CEB1X9 46237042 Ki = 2495 nM T13201 C1VIK9 46237043 Ki = 101 nM T13201 C3RJ5M 46237044 Ki = 4260 nM T13201 CU5Y9E 46237045 Ki = 3830 nM T13201 CM7N6J 46237172 Ki = 737 nM T13201 CP15GJ 46237173 Ki = 9.4 nM T13201 C25FBC 46567082 Ki = 76.8 nM T13201 CQN8K4 46635132 Ki = 658.9 nM T13201 CA4FJ2 46703925 Ki = 6530 nM T13201 C2WB4C 46703927 Ki = 8840 nM T13201 CO2IU4 46704079 Ki = 1520 nM T13201 CB85EQ 46704080 Ki = 78 nM T13201 CAE9Z3 46704081 Ki = 101 nM T13201 CD5V6T 46704082 Ki = 8900 nM T13201 CQ0YA8 46830113 Ki = 630 nM T13201 CEJ2L7 46830114 Ki = 1000 nM T13201 C5MB8F 46845029 IC50 = 9100000 nM T13201 C8MR0H 46847340 IC50 = 380 nM T13201 CRS8J6 46860267 Ki = 89.2 nM T13201 C2RA7G 46861342 Ki = 16.1 nM T13201 C2S4YC 46866644 IC50 = 980 nM T13201 C7QR8Y 46866645 IC50 = 710 nM T13201 CUH07J 46866646 IC50 = 750 nM T13201 C8GK4C 46866647 IC50 = 520 nM T13201 CT65RE 46868356 Ki = 4140 nM T13201 C7CQ6I 46871755 Ki = 27 nM T13201 CNEO10 46871889 Ki = 920 nM T13201 C7UKN2 46884029 Ki = 110 nM T13201 C1DCM9 46884093 Ki = 2400 nM T13201 C4ALG9 46884132 Ki = 81 nM T13201 CTRY21 46884169 Ki = 110 nM T13201 CBM20W 46884215 Ki = 3210 nM T13201 CR61DW 46884254 Ki = 97 nM T13201 CH14SG 46884922 Ki = 510 nM T13201 CFK1L8 46884953 Ki = 930 nM T13201 C9QVN3 46884954 Ki = 680 nM T13201 C60IQZ 46888469 IC50 = 12100000 nM T13201 CD4LT3 46888470 IC50 = 10230000 nM T13201 CW94IO 46888471 IC50 = 11230000 nM T13201 CE19LY 46888472 IC50 = 10700000 nM T13201 C2X6AE 46888473 IC50 = 13710000 nM T13201 C0AN1G 46890958 Ki = 23 nM T13201 C08WJF 46890959 Ki = 22 nM T13201 C9UK8S 46891017 Ki = 22 nM T13201 C2KT4I 46891018 Ki = 43000 nM T13201 C93AIR 46899573 Ki = 122000 nM T13201 C4GZ6A 46907387 Ki = 6670 nM T13201 CJ0R2O 46911381 Ki = 340 nM T13201 C6YK2E 46913624 Ki = 3560 nM T13201 CAF1K0 46913625 Ki = 36400 nM T13201 CO60NB 46918149 Ki = 2170 nM T13201 C9T3WF 46933594 Ki = 5880 nM T13201 C1WE2D 46933744 Ki = 1130 nM T13201 CUHI56 46933745 Ki = 1170 nM T13201 C27DFQ 46933746 Ki = 1180 nM T13201 CSQG87 46933747 Ki = 1090 nM T13201 C08BKN 46933748 Ki = 1100 nM T13201 C54PRX 46933749 Ki = 14200 nM T13201 CP62AV 46933896 Ki = 12100 nM T13201 C03FQY 46943413 Ki = 843 nM T13201 C31ZQL 49843495 Ki = 781 nM T13201 CQJX35 49843496 Ki = 427 nM T13201 CQA97T 49844531 IC50 = 50 nM T13201 CN2U1Z 49844532 IC50 = 70 nM T13201 C5SWC2 49844677 Ki = 460 nM T13201 CD73OF 49844678 Ki = 740 nM T13201 C56KLI 49844679 IC50 = 90 nM T13201 CR87DE 49844829 IC50 = 130 nM T13201 CCOB94 49929067 Ki = 37.9 nM T13201 CY45IU 49957432 IC50 = 266.56 nM T13201 C5Z2QA 50741845 Ki > 50000 nM T13201 CVC35K 50899076 IC50 = 7820 nM T13201 CR3I2H 50899077 IC50 = 9430 nM T13201 CEHP41 50909907 Ki = 23.4 nM T13201 CB4O0Y 50909908 Ki = 9 nM T13201 CU9S2J 50939824 Ki = 3465 nM T13201 CCM82N 50939825 Ki = 235 nM T13201 C1QBZ3 50942416 Ki = 11.3 nM T13201 C62ZDQ 51035422 Ki = 1098 nM T13201 CW0CJ2 51035423 Ki = 3075 nM T13201 C5CR2F 51039206 Ki = 970 nM T13201 C3SH7R 51039207 Ki = 5660 nM T13201 CS5ZR3 51039209 Ki = 1190 nM T13201 C8TR3Z 51047320 Ki = 42.5 nM T13201 CHK5G9 51059586 Ki > 50000 nM T13201 CDP03R 51076628 Ki = 0.5645 nM T13201 C5BA0P 51346838 Ki = 5246 nM T13201 C8G3WE 51346839 Ki = 4382 nM T13201 C8XGV5 51349458 Ki = 4610 nM T13201 C4S5NC 51349459 Ki = 3360 nM T13201 CZH4T2 51349599 Ki = 5640 nM T13201 CK3U6Q 51349600 Ki = 860 nM T13201 CDF2V8 51349601 Ki = 12600 nM T13201 CG26DK 51349604 Ki = 8750 nM T13201 CUP39M 51355749 Ki = 536 nM T13201 CJ1M5T 51355750 Ki = 57 nM T13201 CBL9U1 51356010 Ki = 1170 nM T13201 CLG43P 51669707 IC50 = 8240 nM T13201 C1FM4S 52940811 Ki = 2169 nM T13201 CE15GD 52941031 Ki = 781 nM T13201 CE7WD6 52942084 Ki = 1736 nM T13201 CRMY05 52942168 Ki = 2131 nM T13201 C7OA0E 52942246 Ki = 3924 nM T13201 C4O3HF 52942279 Ki = 1290 nM T13201 C2OQL5 52942476 Ki > 100000 nM T13201 C0R5HD 52943223 Ki = 7085 nM T13201 CCNT92 52943270 Ki = 1751 nM T13201 CXMY91 52943276 Ki = 5412 nM T13201 CC67HN 52943455 Ki = 2151 nM T13201 C50ELG 52943614 Ki > 100000 nM T13201 C7HU5Q 52944525 Ki > 10000 nM T13201 CB4UY1 52944603 Ki = 1691 nM T13201 C3G6WM 52944864 Ki > 100000 nM T13201 C20FAL 52945268 Ki = 6135 nM T13201 C3MLZ1 52945326 Ki = 4424 nM T13201 CBGN39 52945721 Ki = 1435 nM T13201 CCV6U5 52945740 Ki = 5853 nM T13201 CX28EM 52945837 Ki = 27400 nM T13201 C6ZCQ2 52947045 Ki = 479 nM T13201 CRVI93 52948047 Ki > 100000 nM T13201 CDNI78 52948211 Ki = 5940 nM T13201 CAW78K 52948213 Ki = 2489 nM T13201 CA59GT 52948974 Ki = 5542 nM T13201 C14WUN 52949402 Ki = 6799 nM T13201 CW92IL 52949544 Ki = 1460 nM T13201 CLK0S1 52950139 Ki = 8170 nM T13201 CPGW70 53245686 Ki = 40 nM T13201 CF89ML 53307609 Ki = 43510 nM T13201 C60FVH 53317618 Ki = 1042 nM T13201 C7FJN3 53318913 Ki = 920 nM T13201 CPSU85 53320228 Ki = 5513 nM T13201 C6VN4G 53320229 Ki = 81.5 nM T13201 CKRO12 53321135 Ki = 5960 nM T13201 CTF92V 53322463 Ki = 1180 nM T13201 CQ8R0Y 53322880 Ki = 1241 nM T13201 CA80RT 53322881 Ki = 3130 nM T13201 CTMG14 53322882 Ki = 9711 nM T13201 C8Z2IL 53324362 Ki = 4500 nM T13201 C9PDY6 53326762 Ki = 4964 nM T13201 CK4ZG3 53342705 Ki = 0.885 nM T13201 CHF62Q 53361485 IC50 = 6800 nM T13201 CJ3F4R 53361486 IC50 = 1750 nM T13201 C08REF 53364160 Ki = 420 nM T13201 C32UEX 53364161 Ki = 420 nM T13201 CHWX25 53364162 Ki = 9703 nM T13201 C58YMC 53371608 Ki = 6125 nM T13201 C0NUM6 53386724 Ki = 512 nM T13201 C54FGU 53386866 Ki = 311 nM T13201 CRI54V 53386867 Ki = 714 nM T13201 CUX7S4 53386868 Ki = 692 nM T13201 CSA60L 53389267 Ki = 50.1 nM T13201 C8VXD9 53389268 Ki = 42.5 nM T13201 CV40HR 53426278 Ki = 340 nM T13201 CUI84R 53439104 Ki = 700 nM T13201 C6T5RC 53483944 Ki = 78 nM T13201 CM5KX6 53483945 Ki = 76 nM T13201 C3M4EL 53483958 Ki = 416000 nM T13201 CCFP92 53516400 Ki = 18.5 nM T13201 CY2MI0 54077127 Ki > 10000 nM T13201 CB6W4D 54577841 Ki > 10000 nM T13201 CI83DC 54578707 Ki = 736.5 nM T13201 CHCT45 54580732 Ki = 41 nM T13201 CEAP89 54581017 Ki = 380000 nM T13201 CYB47X 54581736 Ki = 43 nM T13201 CJI09P 54582050 Ki = 420000 nM T13201 CW2KI4 54582723 Ki = 32 nM T13201 CWK6B0 54582724 Ki = 950 nM T13201 CBS8R1 54584666 Ki = 137 nM T13201 CJ3UE2 54584667 Ki = 395 nM T13201 C69YAR 54584941 Ki = 104000 nM T13201 CO0BD9 54585508 Ki = 587 nM T13201 C0A5OZ 54612935 Ki = 7.9 nM T13201 C6SM5T 54613427 Ki = 1540 nM T13201 C6X7QG 54613732 Ki = 92.7 nM T13201 CKB0G9 54669765 Ki = 112 nM T13201 CS8IV7 54669781 Ki = 119 nM T13201 C0PJ1K 54677403 Ki > 10000 nM T13201 CAS91K 54682930 Ki = 95000 nM T13201 CQ3XK0 54758050 Ki = 115 nM T13201 C5ON9E 54758136 Ki = 103 nM T13201 C0K2LN 54758137 Ki = 4070 nM T13201 C5Q9XC 54758138 Ki = 101 nM T13201 CLT0W2 54758232 Ki = 184 nM T13201 C5V4GI 54758233 Ki = 119 nM T13201 C98JVL 54758234 Ki = 3920 nM T13201 CXBF42 54758235 Ki = 3730 nM T13201 C4EL5V 54758236 Ki = 142 nM T13201 CU19DH 54758322 Ki = 632 nM T13201 CE53AN 54758323 Ki = 105 nM T13201 CK3Q0O 54758324 Ki = 6860 nM T13201 CE2O3A 54768697 Ki = 2460 nM T13201 C5SB4M 54768698 Ki = 5380 nM T13201 CBNP25 54768699 Ki = 251000 nM T13201 C9Z4RJ 54772055 Ki = 7600 nM T13201 CB3EC8 54772057 Ki = 5450 nM T13201 CE6LD4 54772059 Ki = 4560 nM T13201 CD5P1I 54772061 Ki = 2910 nM T13201 C3RQX8 54940826 Ki = 617 nM T13201 C0ZJ2L 55629711 Ki = 83.8 nM T13201 CGR24P 56659114 Ki = 300 nM T13201 CRHT26 56659115 Ki = 45 nM T13201 CD56GS 56659116 Ki = 450 nM T13201 CK89GH 56659335 Ki = 502 nM T13201 C05JRQ 56659336 Ki = 1659 nM T13201 CEC29W 56659337 Ki = 2040 nM T13201 C2TW1F 56659553 Ki = 91 nM T13201 CO9SW8 56659554 Ki = 6390 nM T13201 CVRM21 56659555 Ki = 3.2 nM T13201 CJ43WP 56659826 Ki = 91900 nM T13201 CP5QI2 56662619 Ki = 43 nM T13201 CZ4HI1 56662794 Ki = 109 nM T13201 CD8SR3 56662795 Ki = 1245 nM T13201 CF0J6I 56663002 Ki = 96 nM T13201 CH0MV2 56663442 Ki = 5650 nM T13201 CM07OK 56663443 Ki = 78 nM T13201 C6M0HP 56666075 Ki = 39 nM T13201 CVM8W4 56666268 Ki = 4550 nM T13201 C89SEG 56666269 Ki = 2360 nM T13201 C36TYE 56666270 Ki = 3704 nM T13201 CD5OZ4 56666482 Ki = 94 nM T13201 CI93KS 56666719 Ki = 65800 nM T13201 CKT5V0 56669476 Ki = 35 nM T13201 C9NV7U 56669478 Ki = 32 nM T13201 CR9F8U 56670316 Ki = 87 nM T13201 CF1J7H 56670317 Ki = 674000 nM T13201 CWNF20 56673403 Ki = 3650 nM T13201 CT29KP 56673404 Ki = 6340 nM T13201 C7DU3M 56673405 Ki = 6.8 nM T13201 CHV04E 56673655 Ki = 9530 nM T13201 C4YI1B 56673656 Ki = 75400 nM T13201 CKL09N 56673817 Ki = 102 nM T13201 C8SY2J 56676310 Ki = 40 nM T13201 CI2R9B 56676517 Ki = 673 nM T13201 C9X7VM 56676518 Ki = 1324 nM T13201 CF86WB 56676713 Ki = 5.1 nM T13201 CDH07V 56677155 Ki = 5590 nM T13201 CR7D6S 56677156 Ki = 806000 nM T13201 CSKB42 56679637 Ki = 27 nM T13201 C2U1VF 56679839 Ki = 607 nM T13201 CS81JH 56680034 Ki = 3870 nM T13201 C02WBE 56680461 Ki = 62 nM T13201 C7D2IN 56682958 Ki = 30 nM T13201 CGX98C 56682960 Ki = 40 nM T13201 C2UE8F 56682961 Ki = 36 nM T13201 CEZ3F5 56683163 Ki = 3472 nM T13201 C4LB1M 56683164 Ki = 3021 nM T13201 CZS9V5 56683165 Ki = 1549 nM T13201 C8V1PA 56683626 Ki = 8637 nM T13201 CXL7Q1 56683627 Ki > 50000 nM T13201 CIJ9V0 56684131 Ki = 155 nM T13201 CTWZ62 56836370 Ki = 373 nM T13201 C49PBJ 56836371 Ki = 569 nM T13201 CK7Y8J 56836443 Ki = 2590 nM T13201 CY7Z1A 56836444 Ki = 1560 nM T13201 CV0ST7 56836445 Ki = 363 nM T13201 C0O3UI 56836446 Ki = 395 nM T13201 C0PKB5 56836447 Ki = 484 nM T13201 CZ9F7P 56836511 Ki = 158 nM T13201 COY29V 56836512 Ki = 747 nM T13201 C7PWG1 56836513 Ki = 307 nM T13201 C4CF8M 56836514 Ki = 192 nM T13201 C4IRK8 56836515 Ki = 538 nM T13201 CH52DA 56921864 Ki = 2260 nM T13201 C0Z8WY 56925533 Ki = 880 nM T13201 CTFL92 56928044 Ki = 681 nM T13201 CC3Q9S 56928516 Ki = 5962 nM T13201 CO18AP 57011620 Ki = 110 nM T13201 C4VGE9 57047254 Ki = 34.3 nM T13201 CNG76Q 57326130 Ki = 4.8 nM T13201 C81YCD 57326131 Ki = 33.5 nM T13201 C4TV1U 57326132 Ki = 21.1 nM T13201 CHL0B3 57326133 Ki = 31.8 nM T13201 C5Z4SW 57326134 Ki = 31.9 nM T13201 CFU62Y 57326227 Ki = 4.5 nM T13201 C97HYX 57326228 Ki = 8.6 nM T13201 CS4I5T 57326229 Ki = 2.5 nM T13201 CUR32K 57334711 Ki = 1040 nM T13201 C2CD1R 57334712 Ki = 1030 nM T13201 C1K0DM 57334713 Ki = 1100 nM T13201 CP7YR5 57345662 Ki = 9 nM T13201 C0S2YZ 57383964 Ki = 6300 nM T13201 C97GHV 57383965 Ki = 4260 nM T13201 CXW5D3 57384052 Ki = 8780 nM T13201 C4XF9A 57384114 Ki = 6040 nM T13201 CS76WU 57384115 Ki = 7500 nM T13201 C0UBL5 57384116 Ki = 7880 nM T13201 C16AGY 57384117 Ki = 4040 nM T13201 CVWK43 57386884 Ki = 8320 nM T13201 CR3C7D 57386885 Ki = 7570 nM T13201 C9CX4B 57386886 Ki = 8180 nM T13201 CZOD69 57386887 Ki = 7170 nM T13201 CZN72E 57386888 Ki = 9240 nM T13201 C9JU0H 57386889 Ki = 8510 nM T13201 CQ0I4V 57386890 Ki = 66300 nM T13201 C8Z0DJ 57387135 Ki = 42900 nM T13201 C1HZS5 57387136 Ki = 38800 nM T13201 C7EN6Z 57387137 Ki = 91700 nM T13201 C87ASQ 57387395 Ki = 950000 nM T13201 CQW5T3 57387397 Ki = 124000 nM T13201 CT3B0Z 57387636 Ki = 7600 nM T13201 CV4C7B 57390570 Ki = 101 nM T13201 CS5O2D 57390571 Ki = 957 nM T13201 C14VNC 57390572 Ki = 5213 nM T13201 C09GQI 57392249 Ki = 4930 nM T13201 CY81SU 57392250 Ki = 6410 nM T13201 CMEV16 57392251 Ki = 3720 nM T13201 C94YIX 57392252 Ki = 7680 nM T13201 CDP3C2 57392352 Ki = 3514 nM T13201 C13FJU 57392368 Ki = 1120 nM T13201 CM7S3H 57394009 Ki = 3770 nM T13201 CHAF57 57394010 Ki = 2940 nM T13201 CV7K9Y 57394771 Ki = 6840 nM T13201 CM4SL9 57394772 Ki = 7980 nM T13201 C1M0LS 57394809 Ki = 540 nM T13201 CJ5XK2 57395770 Ki = 5510 nM T13201 CV6QX4 57395771 Ki = 100 nM T13201 CP9D5B 57395861 Ki = 4790 nM T13201 CY5G4Z 57395885 Ki = 2450 nM T13201 C5RX6H 57396029 Ki = 12920 nM T13201 CHG91B 57396529 Ki = 5790 nM T13201 C9H4VS 57396530 Ki = 110 nM T13201 C6XD2O 57397549 Ki = 4570 nM T13201 C64VIW 57397550 Ki = 5900 nM T13201 CR30XN 57397648 Ki = 995 nM T13201 CP75OF 57397664 Ki = 193240 nM T13201 CUAG84 57397836 Ki = 187130 nM T13201 CW43HV 57397837 Ki = 13270 nM T13201 CRIU35 57398318 Ki = 4780 nM T13201 CN6TU2 57398319 Ki = 100 nM T13201 C97OJM 57399231 Ki = 100 nM T13201 C7XAZ3 57399232 Ki = 3770 nM T13201 CK24NA 57399233 Ki = 9 nM T13201 C1MCW8 57399336 Ki = 292109 nM T13201 C2CAM1 57399491 Ki = 10540 nM T13201 CQD65L 57401080 Ki = 5134 nM T13201 C1SK7F 57401081 Ki = 4793 nM T13201 CG3X4V 57401764 Ki = 4060 nM T13201 C4V5KY 57402747 Ki = 6710 nM T13201 CRU53E 57402748 Ki = 6340 nM T13201 C52TUM 57402749 Ki = 100 nM T13201 CQ9ZG2 57402750 Ki = 110 nM T13201 CI3L9R 57402843 Ki = 6003 nM T13201 CW10QX 57402844 Ki = 4815 nM T13201 C80WTZ 57403496 Ki = 6420 nM T13201 CDIM87 57403497 Ki = 7920 nM T13201 C76ZDS 57404539 Ki = 483 nM T13201 CKID78 57411990 Ki = 77 nM T13201 C4ZYF3 57411991 Ki = 68 nM T13201 CDG6R4 57411992 Ki = 32 nM T13201 CKPS17 57411993 Ki = 33 nM T13201 CV13LT 57411994 Ki = 377 nM T13201 CW1TU4 57412422 Ki = 514 nM T13201 CT4BV9 57412423 Ki = 50.4 nM T13201 C31NWX 57412424 Ki = 24.6 nM T13201 CD86ER 57412425 Ki = 1050 nM T13201 CB94YU 57412426 Ki = 83.1 nM T13201 C2K8YJ 57412507 Ki = 9.2 nM T13201 CSF4V6 57412508 Ki = 667 nM T13201 CHAO86 57412509 Ki = 72.3 nM T13201 C3U6TH 57412510 Ki = 24.3 nM T13201 C40LOS 57412511 Ki = 1210 nM T13201 CZ47VT 57412512 Ki = 4165 nM T13201 C28WRD 57412600 Ki = 474 nM T13201 C2XPG5 57413583 Ki = 6.7 nM T13201 CM2AY7 57413584 Ki = 6.7 nM T13201 C5JDQ1 57413825 Ki = 3203 nM T13201 C5M4CN 57413826 Ki = 101 nM T13201 C3D7KS 57413827 Ki = 107 nM T13201 CJO26X 57413828 Ki = 79 nM T13201 CA4CD7 57413968 Ki = 9576 nM T13201 CQ1ZK6 57519697 Ki = 1130 nM T13201 CX8W0C 57624955 IC50 = 4800 nM T13201 CG3W0D 58404071 Ki = 850 nM T13201 CT3B7P 58477593 Ki = 296 nM T13201 C01TQW 59079460 Ki = 62.2 nM T13201 CF1NG0 60155028 Ki = 1.186 nM T13201 C0PRW7 60155029 Ki = 1.176 nM T13201 CNX97Q 60155030 Ki = 1.262 nM T13201 CR0Z7W 60155031 Ki = 0.994 nM T13201 CI2WL7 60155120 Ki = 1.131 nM T13201 CM57BF 60155121 Ki = 0.896 nM T13201 C5VF9X 60155122 Ki = 1.544 nM T13201 C2U8VH 60155123 Ki = 0.993 nM T13201 CNR53M 60155124 Ki = 12500 nM T13201 CYQM98 60201413 Ki = 1425 nM T13201 CGWU14 60201414 Ki = 72 nM T13201 C6TP2W 60201415 Ki = 633 nM T13201 C1JVP9 60201416 Ki = 148 nM T13201 CQZN79 60201417 Ki = 43 nM T13201 CVU0B4 60201577 Ki = 473 nM T13201 CS3N6M 60201578 Ki = 237 nM T13201 CB45GM 60201579 Ki = 379 nM T13201 C9V6EY 60446869 Ki = 913.4 nM T13201 COW0X5 61580695 Ki = 92.1 nM T13201 C1CVG9 61580845 Ki = 5.3 nM T13201 C9UD2V 62141270 Ki = 2078 nM T13201 CZ4BQ6 66571808 Ki > 10000 nM T13201 CGB46T 66571809 Ki > 10000 nM T13201 CT0S3A 66572208 Ki > 10000 nM T13201 C2J7GW 66572313 Ki = 57870 nM T13201 C7J5RN 66573254 Ki = 93420 nM T13201 CGF3W6 66586679 Ki = 920 nM T13201 CN84CU 66586879 Ki = 970 nM T13201 CAD3V2 67662627 Ki = 7181 nM T13201 C54HCL 68341722 Ki > 10000 nM T13201 C4MB5P 68602550 Ki > 10000 nM T13201 CA7F0J 68819643 Ki = 1509 nM T13201 CV6PY2 68833705 Ki = 3499 nM T13201 C23JZS 70037678 Ki = 44.2 nM T13201 C6RVC3 70202738 Ki = 320.4 nM T13201 C3BYV1 70681295 IC50 = 46200 nM T13201 CDO92J 70681983 Ki = 1.123 nM T13201 CHC54M 70681984 Ki = 0.821 nM T13201 C1FY3K 70681985 Ki = 1.092 nM T13201 CSW7I0 70681986 Ki = 1.077 nM T13201 CP65RU 70681987 Ki = 0.694 nM T13201 CFT68C 70681988 Ki = 1.092 nM T13201 C2Y5KV 70682044 Ki = 3000 nM T13201 CR0D9S 70684100 Ki = 1.089 nM T13201 CRZ8S1 70684101 Ki = 1.123 nM T13201 COS95H 70684102 Ki = 1.115 nM T13201 CT5PH1 70684103 Ki = 0.758 nM T13201 C4SX6F 70685487 IC50 = 9070 nM T13201 C9P4BK 70685635 Ki = 48.4 nM T13201 C5XTY9 70686245 Ki = 1.155 nM T13201 C5A6TI 70687643 IC50 = 5850 nM T13201 CPD1N7 70688361 Ki = 0.699 nM T13201 C4L2OE 70688362 Ki = 0.52 nM T13201 CZO9C5 70688363 Ki = 0.537 nM T13201 CAD39I 70688364 Ki = 0.75 nM T13201 CRHL03 70689373 Ki = 43 nM T13201 CVQ6B2 70689703 IC50 = 8120 nM T13201 C9G7QF 70689704 IC50 = 8300 nM T13201 C7N4RT 70690386 Ki = 1.142 nM T13201 CQD8R9 70690387 Ki = 0.977 nM T13201 C1T4JL 70690936 Ki = 4020 nM T13201 CUY3O8 70690937 Ki = 1650 nM T13201 C5C9SL 70691832 IC50 = 54100 nM T13201 CP81SC 70691833 IC50 = 9720 nM T13201 CQR91N 70692438 Ki = 41360 nM T13201 CXF59L 70692549 Ki = 1.311 nM T13201 CV76WB 70692550 Ki = 1.244 nM T13201 C89LCZ 70692551 Ki = 0.694 nM T13201 C1K8VS 70692552 Ki = 1.49 nM T13201 CO5JP7 70692553 Ki = 1.162 nM T13201 CK5Y7G 70692554 Ki = 0.811 nM T13201 CGD06J 70692555 Ki = 1.241 nM T13201 C5QOK4 70692556 Ki = 1.143 nM T13201 CF0YQ6 70693894 IC50 = 7100 nM T13201 C4BDK3 70694601 Ki = 1.244 nM T13201 CW8YA7 70694602 Ki = 0.611 nM T13201 CCYE61 70694603 Ki = 1.112 nM T13201 CEF1J8 70694604 Ki = 0.818 nM T13201 C4C0HK 70694605 Ki = 1.237 nM T13201 CBDQ72 70694606 Ki = 1 nM T13201 C95YWO 70695124 Ki = 6200 nM T13201 CSH7P1 70696148 Ki = 157 nM T13201 CWJ0Q8 70696540 Ki = 25341 nM T13201 CWSA94 70696638 Ki = 1.149 nM T13201 CREC06 70696639 Ki = 1.118 nM T13201 CJ4M9S 70696640 Ki = 0.901 nM T13201 CHFY23 70696641 Ki = 0.998 nM T13201 C3Z7ER 70696642 Ki = 0.679 nM T13201 C6E4UW 70696643 Ki = 0.978 nM T13201 C0SP9E 70696644 Ki = 0.98 nM T13201 CAFH02 70696645 Ki = 1.054 nM T13201 CWQM13 70696646 Ki = 0.75 nM T13201 CNS4U0 70791951 Ki = 557 nM T13201 CS58EL 70792049 Ki = 487 nM T13201 C8FB0P 71273627 Ki = 0.712 nM T13201 CJH6Y7 71273628 Ki = 0.81 nM T13201 CXG0H9 71273629 Ki = 1 nM T13201 CUT6R1 71273630 Ki = 0.709 nM T13201 CH49BT 71273631 Ki = 0.774 nM T13201 CK2U8R 71273632 Ki = 1.337 nM T13201 C2F9PC 71273633 Ki = 1.071 nM T13201 CV8FW3 71273635 Ki = 0.612 nM T13201 CQJ61A 71273738 Ki = 1.031 nM T13201 CSMV41 71273739 Ki = 1.034 nM T13201 CYW59B 71273740 Ki = 1.058 nM T13201 CU0KV6 71273743 Ki = 1.236 nM T13201 CC21VR 71273744 Ki = 1.225 nM T13201 C80KUG 71273750 Ki = 1.446 nM T13201 CJHN78 71415156 Ki = 437 nM T13201 C8NYL3 71449075 Ki = 39 nM T13201 CRN2O1 71449118 Ki = 108 nM T13201 C16PMU 71449958 IC50 = 9700 nM T13201 CXJ16H 71450117 Ki = 193 nM T13201 CR79UB 71450332 Ki = 2437 nM T13201 C09RTJ 71450813 Ki = 930 nM T13201 C6VQI7 71450814 Ki = 680 nM T13201 CK04AG 71450862 Ki = 40 nM T13201 CU3XD2 71450931 Ki = 29 nM T13201 C72GOW 71450940 Ki = 350 nM T13201 CT8E7N 71451561 Ki = 241 nM T13201 CHI2Z6 71452138 Ki = 224 nM T13201 CNI0R5 71452603 Ki = 774 nM T13201 C9D3CU 71452683 Ki = 510 nM T13201 C4E6PS 71453593 IC50 = 620 nM T13201 CP27AT 71453970 Ki = 1573 nM T13201 CW49YT 71453971 Ki = 235 nM T13201 C52WNJ 71454366 Ki = 2496 nM T13201 CT90CD 71454373 Ki = 112.3 nM T13201 CKB14Q 71454522 Ki = 240 nM T13201 CZ0P8A 71454523 Ki = 54 nM T13201 CB8JA3 71455488 Ki = 318 nM T13201 C02UHX 71455489 Ki = 65 nM T13201 CZ0S7D 71455712 Ki = 3106 nM T13201 CUX07I 71455715 Ki = 1883 nM T13201 C9COK3 71456113 Ki = 4065 nM T13201 CICJ97 71457274 Ki = 212 nM T13201 CL2BN6 71457492 Ki = 580 nM T13201 C4L0BG 71457918 Ki = 1925 nM T13201 C0XQ5P 71457958 Ki = 750 nM T13201 CSD08X 71458070 Ki = 105 nM T13201 CWHN25 71459359 Ki = 583 nM T13201 CE31LC 71459360 Ki = 4790 nM T13201 C7G6IR 71459681 Ki = 31700000 nM T13201 C70MBK 71459826 Ki = 4830 nM T13201 C95MKT 71459827 Ki = 3742 nM T13201 C5WYI8 71459828 Ki = 899 nM T13201 CX9KJ3 71459903 Ki = 350 nM T13201 CO30KR 71459904 Ki = 1200 nM T13201 CJX65D 71459953 Ki = 205 nM T13201 C14NRE 71459973 Ki = 1000 nM T13201 CD93TU 71461134 Ki = 776 nM T13201 C3WKX5 71461135 Ki = 4563 nM T13201 C3YSR8 71461136 Ki = 1571 nM T13201 CS1WI7 71461542 Ki = 3613 nM T13201 C7VQ1R 71461543 Ki = 3217 nM T13201 C4X1BZ 71462495 IC50 = 9740 nM T13201 CUM2H8 71462868 Ki = 4364 nM T13201 CU4N0L 71462869 Ki = 3226 nM T13201 C9KZA2 71462872 Ki = 4065 nM T13201 CI6V9W 71489159 Ki = 4310 nM T13201 CDQ8Z3 71498310 IC50 = 60.46 nM T13201 CIE7T0 71498311 IC50 = 1341.59 nM T13201 CN6K9Q 71498738 IC50 = 1541.18 nM T13201 CX6JP1 71498761 IC50 = 772.88 nM T13201 C98SLI 71498762 IC50 = 866.74 nM T13201 CJ2TX7 71498763 IC50 = 664.71 nM T13201 C0QX8S 71498764 IC50 = 44.38 nM T13201 CQPM90 71508409 Ki = 102 nM T13201 C8CH5R 71508458 Ki = 219 nM T13201 CF4RQ9 71508459 Ki = 62.3 nM T13201 CJ5KW8 71508507 Ki = 115 nM T13201 C0VWD1 71508508 Ki = 1278 nM T13201 CHZ93F 71508509 Ki = 485 nM T13201 CLD8G6 71508510 Ki = 490 nM T13201 C58ZQR 71508548 Ki = 384 nM T13201 CBP08O 71508550 Ki = 806 nM T13201 CMHG14 71521493 Ki = 5700 nM T13201 CHN53G 71521494 Ki = 5100 nM T13201 CZJ5M6 71521495 Ki = 9300 nM T13201 CFBE53 71521496 Ki = 6800 nM T13201 CME27W 71521497 Ki = 3600 nM T13201 C24XWU 71521575 Ki = 8500 nM T13201 CJF68W 71521576 Ki = 5500 nM T13201 CHL8P3 71522144 Ki = 6780 nM T13201 CEYG83 71522162 Ki = 92000 nM T13201 CZ78YT 71522163 Ki > 100000 nM T13201 C8NAF3 71545047 Ki = 6860 nM T13201 C4H6PD 71545048 Ki = 8050 nM T13201 CQ20AS 71545049 Ki = 8880 nM T13201 CG2CL6 71545050 Ki = 6000 nM T13201 C1MET8 71545051 Ki = 7200 nM T13201 CILC35 71545052 Ki = 8110 nM T13201 CGQ97W 71545216 Ki = 8430 nM T13201 C71UMX 71545217 Ki = 8930 nM T13201 C3KJ6D 71545218 Ki = 6710 nM T13201 C0JNF3 71545219 Ki = 7470 nM T13201 CC5EB7 71570660 Ki = 222.48 nM T13201 CA82YW 71570661 Ki = 23.48 nM T13201 CNL58G 71570662 Ki = 225.58 nM T13201 CQKG46 71578358 Ki = 9310 nM T13201 CV6FW1 71578359 Ki = 6720 nM T13201 CDA18G 71578360 Ki = 8300 nM T13201 C3P8YG 71578361 Ki = 10230 nM T13201 CDGY15 71578422 Ki = 51.4 nM T13201 CA5M6S 71578423 Ki = 31.2 nM T13201 CGOR42 71578424 Ki = 48.5 nM T13201 C45YXJ 71578425 Ki = 35.8 nM T13201 C1CKL6 71578426 Ki = 26.5 nM T13201 CR38IX 71578427 Ki = 7.2 nM T13201 CQ8Z5T 71578500 Ki = 25.6 nM T13201 CZ1R3F 71578570 Ki = 52.4 nM T13201 CV0G1A 71578571 Ki = 18.7 nM T13201 CX7T2V 71578640 Ki = 116 nM T13201 COT80J 71578641 Ki = 87 nM T13201 CGV68Z 71578723 Ki = 2644 nM T13201 C7U0LV 71578724 Ki = 1710 nM T13201 C8M0YB 71578725 Ki = 1168 nM T13201 C4F0HB 71578726 Ki = 5932 nM T13201 CZ29IK 71578808 Ki = 3204 nM T13201 C8HMK5 71578809 Ki = 2786 nM T13201 CMH2W4 71578810 Ki = 2046 nM T13201 C7W9BS 71578811 Ki = 77 nM T13201 CU6N9T 71578812 Ki > 10000 nM T13201 CGEJ87 71578813 Ki = 351 nM T13201 C8CM0Q 71578898 Ki = 1197 nM T13201 C19JFD 71578899 Ki = 2120 nM T13201 C0MT2F 71578903 Ki = 1749 nM T13201 CB9R7F 71578904 Ki = 217 nM T13201 C5MLA7 71578977 Ki = 42600 nM T13201 C03THE 71578978 Ki = 39300 nM T13201 CR57YV 71578979 Ki = 41700 nM T13201 CVTN91 71578980 Ki = 175 nM T13201 CBJ18U 71578981 Ki = 7136 nM T13201 CCKJ51 71578982 Ki = 174 nM T13201 C0TKR8 71579053 Ki = 5626 nM T13201 CX4D6V 71579054 Ki = 5179 nM T13201 CJ0UP9 71579055 Ki = 151 nM T13201 CREN23 71579056 Ki = 6764 nM T13201 CP61GE 71579057 Ki = 4224 nM T13201 CXD68U 71579058 Ki = 6796 nM T13201 C19OIY 71579130 Ki = 500 nM T13201 CV0LU6 71602117 Ki = 390 nM T13201 CCE15B 71602410 Ki = 176 nM T13201 CCB72P 71602411 Ki = 33.9 nM T13201 CHL16T 71602412 Ki = 21.8 nM T13201 C2UQV5 71602471 Ki = 22.2 nM T13201 C8K1YM 71602472 Ki = 21.2 nM T13201 CZL96Y 71602476 Ki = 427 nM T13201 CE70AQ 71602537 Ki = 403 nM T13201 C3KPA8 71602538 Ki = 489 nM T13201 CO6FJ4 71602539 Ki = 262 nM T13201 CQ17LM 71602540 Ki = 142.9 nM T13201 C78LKP 71607884 IC50 > 10000 nM T13201 COVC80 71607885 IC50 > 10000 nM T13201 C1MOS8 71607912 IC50 = 220.2 nM T13201 CE0F4T 71607913 IC50 > 10000 nM T13201 CO2LM4 71607914 IC50 > 10000 nM T13201 CNBK57 71607915 IC50 > 10000 nM T13201 CXPO21 71607916 IC50 > 10000 nM T13201 CU24SZ 71607951 IC50 = 85.7 nM T13201 CJQW86 71607952 IC50 > 10000 nM T13201 CR7BQ5 71607953 IC50 > 10000 nM T13201 CPM89A 71607954 IC50 > 10000 nM T13201 C1OPS4 71658869 Ki = 1820 nM T13201 CN2FZ3 71659103 Ki = 250 nM T13201 CC0EU9 71677604 Ki = 428 nM T13201 CS4VW3 71681364 Ki = 532 nM T13201 C5SY2L 71681517 Ki = 45.1 nM T13201 CT1D0W 71681519 Ki = 5.6 nM T13201 CW65GP 71681521 Ki = 6.3 nM T13201 CFS62D 71681523 Ki = 64.1 nM T13201 C96OCT 71681525 Ki = 74.2 nM T13201 C57BRD 71681527 Ki = 81.3 nM T13201 CU45ER 71681529 Ki = 59.1 nM T13201 C7NMJ2 71714066 Ki = 380 nM T13201 C5DEF6 71714067 Ki = 760 nM T13201 C50LSJ 71714068 Ki = 130 nM T13201 C6A1RS 71716868 Ki = 55 nM T13201 C84WSV 71716939 Ki = 93000 nM T13201 CBY8J3 71716994 Ki = 4800 nM T13201 CM4T1R 71717003 Ki = 6550 nM T13201 CN76CQ 71717054 Ki = 2740 nM T13201 CI0SY3 71717570 Ki = 91000 nM T13201 CYGT30 71717571 Ki = 99000 nM T13201 CG4I1X 71718239 Ki = 5100 nM T13201 C4N3VH 71718790 Ki = 0.978 nM T13201 C0LYX1 71718858 Ki = 2980 nM T13201 C4B8KN 71718888 Ki = 134 nM T13201 C7U6NR 71719377 Ki > 100000 nM T13201 CM24ND 71719433 Ki = 720 nM T13201 CT3D5S 71719441 Ki = 4800 nM T13201 CY3CV6 71719496 Ki = 2105 nM T13201 CJG34A 71720036 Ki = 7520 nM T13201 CIU4L2 71720670 Ki = 7400 nM T13201 CN0L8Q 71720672 Ki = 637 nM T13201 CY54DH 71728127 Ki > 10000 nM T13201 C9JAE7 71728128 Ki > 10000 nM T13201 C6HOP3 71728129 Ki > 10000 nM T13201 CRY5D8 71728130 Ki > 10000 nM T13201 CM91JE 71728236 Ki > 10000 nM T13201 C30ZEI 71728237 Ki > 10000 nM T13201 C4JB8W 71728238 Ki > 10000 nM T13201 C5RS9P 71728239 Ki > 10000 nM T13201 CRYC54 71728240 Ki > 10000 nM T13201 C5TKY7 71764398 Ki = 4.8 nM T13201 CMD91U 71764399 Ki = 104 nM T13201 CXO1T9 71764400 Ki = 236 nM T13201 CVEI80 71764401 Ki = 8.6 nM T13201 CVQ1H3 71764402 Ki = 106 nM T13201 CRZ64M 71764403 Ki = 254 nM T13201 CC0X1H 71764607 Ki = 9.8 nM T13201 CK7NI0 71764608 Ki = 4.1 nM T13201 C90YMG 71764609 Ki = 8.5 nM T13201 CK35HL 71764610 Ki = 246 nM T13201 C4SV1I 71764611 Ki = 166 nM T13201 C8NG9B 71764612 Ki = 6.5 nM T13201 CA2M1B 71764613 Ki = 8.7 nM T13201 CR7J6M 71764825 Ki = 4.3 nM T13201 CG09CJ 71764826 Ki = 8.2 nM T13201 CK2N0Z 71764827 Ki = 223 nM T13201 C08RAW 71765040 Ki = 4.9 nM T13201 CGI1J3 71765041 Ki = 7.6 nM T13201 CPT1X2 71765042 Ki = 2.9 nM T13201 C0ROQ1 71770179 Ki = 326 nM T13201 C8W6DJ 71770180 Ki = 444 nM T13201 CB3Y0X 71770181 Ki > 10000 nM T13201 CKHM42 71770182 Ki = 368 nM T13201 CBL41T 71770183 Ki = 150 nM T13201 C30EYH 71770184 Ki = 281 nM T13201 CGA62Y 71770789 Ki = 499 nM T13201 C8GP3J 71770790 Ki = 1434 nM T13201 C04WFV 71770791 Ki = 526 nM T13201 CN4QC0 71770911 Ki = 2540 nM T13201 C6XSA1 71770912 Ki = 746 nM T13201 C5YU4I 71770913 Ki = 750 nM T13201 C4G3HO 71770914 Ki = 3055 nM T13201 CSU93P 71770915 Ki = 2420 nM T13201 C9NAK1 71770916 Ki = 289 nM T13201 C42KOE 71770917 Ki = 2132 nM T13201 CE8IC7 71770918 Ki = 2464 nM T13201 CQJI19 71771031 Ki = 4273 nM T13201 C2ZOB7 71771032 Ki = 709 nM T13201 C93LEJ 71771033 Ki = 224 nM T13201 C5UZM3 71771034 Ki = 7544 nM T13201 CX9N5F 71818212 Ki > 10000 nM T13201 C5IU0Y 72163201 Ki = 432 nM T13201 CNP42E 72163326 Ki = 160 nM T13201 C2KE5D 72163327 Ki = 4260 nM T13201 C0Q5XL 72163343 Ki = 251 nM T13201 C63MIX 72163344 Ki = 185 nM T13201 CL3WV2 72163345 Ki = 340 nM T13201 C4T9DA 72163346 Ki > 10000 nM T13201 CTK07O 72163347 Ki = 770 nM T13201 CE32BF 72163348 Ki = 208 nM T13201 CBN48K 72163465 Ki = 1580 nM T13201 CGB02D 72163466 Ki = 7340 nM T13201 CVFN85 72163467 Ki = 3510 nM T13201 C82RDA 72163468 Ki = 6220 nM T13201 CA1X6Z 72163476 Ki = 143 nM T13201 C7TKJ4 72163610 Ki = 8850 nM T13201 C70OBD 72163611 Ki = 8260 nM T13201 CA0Q4T 72163612 Ki = 2130 nM T13201 C96GMR 72163613 Ki = 9640 nM T13201 CJ2K8R 72163743 Ki = 9490 nM T13201 CPY81U 72163744 Ki = 5330 nM T13201 CC1D3Y 72163745 Ki = 1890 nM T13201 CYH0G5 72163746 Ki = 9340 nM T13201 CEZM40 72163861 Ki = 260 nM T13201 CMBR85 72163862 Ki = 2140 nM T13201 CZ9IE5 72163863 Ki = 3470 nM T13201 CZM75P 72163975 Ki = 4330 nM T13201 CPT0C9 72163976 Ki = 850 nM T13201 C0FM1E 72202020 Ki = 61 nM T13201 CT41SJ 72202021 Ki = 250 nM T13201 CC1SO2 72203951 Ki = 1036.7 nM T13201 CE9Q6G 72203952 Ki = 1646.6 nM T13201 C5YJK2 72203953 Ki = 1239.2 nM T13201 CM2F7D 72204122 Ki = 838.3 nM T13201 C8XDF6 72204123 Ki = 742.3 nM T13201 CO51BD 72204124 Ki = 936.4 nM T13201 CWJE09 72204125 Ki = 1247.9 nM T13201 C8XVK1 72204126 Ki = 1112.5 nM T13201 C7WDI2 72204321 Ki > 10000 nM T13201 CX4G0R 72204928 IC50 > 10000 nM T13201 CG9C6U 72204929 IC50 > 10000 nM T13201 C5A6XZ 72204930 IC50 = 7977 nM T13201 C0XZK4 72204931 IC50 = 6082 nM T13201 C6RY4X 72204933 IC50 = 4570 nM T13201 C4N5AB 72204934 IC50 = 5830 nM T13201 C3H2FZ 72205111 IC50 > 10000 nM T13201 CQ0VX7 72205112 IC50 = 5535 nM T13201 CQ7TI1 72205113 IC50 > 10000 nM T13201 CPAW52 72205114 IC50 > 10000 nM T13201 C2LD3J 72205115 IC50 > 10000 nM T13201 C4E2VS 72543811 Ki > 10000 nM T13201 C3UJ8A 72695827 Ki = 58.5 nM T13201 CX82JD 72696463 Ki = 88 nM T13201 COCV73 72696591 Ki = 203 nM T13201 C5KHD7 72696592 Ki = 238 nM T13201 C4FBA6 72696593 Ki = 90 nM T13201 CO1JM5 72696594 Ki = 81.5 nM T13201 CUF61Q 72696595 Ki = 250 nM T13201 C1SU0Q 72712917 Ki = 4435 nM T13201 COD5F4 72712918 Ki = 9120 nM T13201 CJW7K4 72712919 Ki > 20000 nM T13201 CT2J8A 72712920 Ki > 20000 nM T13201 CRGC51 72713105 Ki = 8718 nM T13201 C61VGR 72713106 Ki = 105 nM T13201 C96WHB 72713107 Ki = 79 nM T13201 CHPN94 72713108 Ki = 84 nM T13201 CJB8R7 72792832 Ki = 2020 nM T13201 C5F7DT 72792833 Ki = 1795 nM T13201 CAC7J8 72792834 Ki = 9226 nM T13201 CFS02B 72792835 Ki = 9441 nM T13201 CF5LW1 72792901 Ki = 9450 nM T13201 C42IFJ 72792902 Ki = 2245 nM T13201 CRMF25 72792903 Ki = 2216 nM T13201 C2G5SR 72792904 Ki = 2936 nM T13201 C6DR9O 72792905 Ki = 9165 nM T13201 CGF5O1 72792967 Ki = 9833 nM T13201 CWH3N9 72792968 Ki = 78.8 nM T13201 C5DSF8 72792969 Ki = 257 nM T13201 C2K6UZ 72792970 Ki = 2130 nM T13201 CGI8K5 72793036 Ki = 3205 nM T13201 C8WO6Z 72793037 Ki = 6452 nM T13201 C6OZ0L 72793038 Ki = 3823 nM T13201 CDTQ64 72793039 Ki = 2351 nM T13201 CY16FM 72793040 Ki = 83.1 nM T13201 CXQN80 72793101 Ki = 73.8 nM T13201 CJ19BH 72793102 Ki = 1876 nM T13201 CO1JT3 73054728 Ki = 245 nM T13201 CA2YM5 73056157 Ki = 134 nM T13201 CXBJ69 73056158 Ki = 185 nM T13201 CT62PI 73056159 Ki = 180 nM T13201 CL8V1X 73056160 Ki = 193 nM T13201 CX5ZV7 73056161 Ki = 151 nM T13201 C1YLW5 73056162 Ki = 132 nM T13201 CL1H0W 73056449 Ki = 247 nM T13201 C0VNX8 73056450 Ki = 91.3 nM T13201 C8Z6YK 73056451 Ki = 130 nM T13201 C0RZW2 73056452 Ki = 367 nM T13201 CR2HU6 73056453 Ki = 162 nM T13201 CI12KH 73056454 Ki = 753 nM T13201 CXHE13 73056743 Ki = 86.4 nM T13201 C3CHO7 73056744 Ki = 390 nM T13201 C3FU9P 73056745 Ki = 16300 nM T13201 C1G8YT 73056746 Ki = 27500 nM T13201 CT2S3D 73056747 Ki = 32800 nM T13201 CM12LF 73056748 Ki = 6540 nM T13201 C4MIP9 73345840 Ki = 327 nM T13201 C4Z7PY 73346473 Ki = 864 nM T13201 C48AKL 73346474 Ki = 2650 nM T13201 CY2AH8 73346475 Ki = 1250 nM T13201 C8QJU7 73346691 Ki = 10 nM T13201 C0PA8K 73346692 Ki = 13 nM T13201 CT6C3G 73346693 Ki = 15 nM T13201 CVN4A3 73346695 Ki = 21 nM T13201 CM9K3D 73346697 Ki = 14 nM T13201 C3Y4VZ 73347324 Ki = 27.8 nM T13201 C1WQ0C 73347968 Ki = 729 nM T13201 CEHI16 73348197 Ki = 51 nM T13201 C18GUI 73348198 Ki > 1000 nM T13201 C3CJ0F 73349055 Ki > 10000 nM T13201 C75IEZ 73349056 Ki > 10000 nM T13201 CK7MD1 73349516 Ki = 397 nM T13201 CJRE74 73349517 Ki = 278 nM T13201 CK98JL 73349518 Ki = 5400 nM T13201 C6S7RY 73349758 Ki = 54 nM T13201 C2JP5U 73349759 Ki = 965.03 nM T13201 CBL42E 73350409 Ki = 24.6 nM T13201 CP3E7Q 73350410 Ki = 23.9 nM T13201 C38QDY 73351066 Ki = 346 nM T13201 COM17Y 73351067 Ki = 4335 nM T13201 CN96PE 73351280 Ki = 62 nM T13201 CX1J7D 73352124 Ki > 10000 nM T13201 CXJL10 73352125 Ki > 10000 nM T13201 CBN25I 73352538 Ki = 169 nM T13201 CRDB68 73352539 Ki = 2450 nM T13201 C4SNT8 73352540 Ki = 5335 nM T13201 C3M2UH 73354029 Ki = 1346 nM T13201 CB7Z2K 73355560 Ki = 438 nM T13201 CR81ON 73355561 Ki = 541 nM T13201 C60FZE 73355562 Ki = 1285 nM T13201 CAK9J2 73355834 Ki = 36 nM T13201 CC2P6U 73356651 Ki > 10000 nM T13201 CC9AE6 73356652 Ki > 10000 nM T13201 C3SB2W 73357104 Ki = 3320 nM T13201 C79KVE 73357105 Ki = 1340 nM T13201 COP7H8 73357339 Ki = 12 nM T13201 CA3YT9 73894059 Ki = 90 nM T13201 C53JCV 74766009 Ki = 86.5 nM T13201 C53PBO 74766010 Ki = 81.3 nM T13201 CLPY57 74766011 Ki = 206 nM T13201 C7EF5V 76310135 Ki = 546 nM T13201 CLX6H0 76310136 Ki = 509 nM T13201 C9K6XP 76310137 Ki = 1347 nM T13201 CX0Y6K 76310141 Ki = 3576 nM T13201 C54AJY 76310148 Ki = 87 nM T13201 CR56JE 76310328 Ki > 100000 nM T13201 CCD80R 76310490 Ki > 10000 nM T13201 CUB9V2 76310833 Ki = 463 nM T13201 C4S3QC 76310834 Ki = 4480 nM T13201 CY7AV1 76310835 Ki = 288 nM T13201 CTJ50C 76310908 Ki > 50000 nM T13201 CEWJ18 76310909 Ki > 50000 nM T13201 CR9G4Q 76311013 Ki = 7.1 nM T13201 CE7O5U 76311014 Ki = 28.4 nM T13201 CV19YL 76311015 Ki = 8.3 nM T13201 CO0PZ4 76311101 Ki > 10000 nM T13201 CGT0J3 76311102 Ki > 10000 nM T13201 CD3LU2 76311370 Ki = 510 nM T13201 C3JCD1 76311371 Ki = 12700 nM T13201 C70UYF 76311372 Ki = 285 nM T13201 C3JFR9 76311373 Ki = 33 nM T13201 C5POS7 76311374 Ki = 400 nM T13201 CI64FZ 76311402 Ki = 1710 nM T13201 CVW59F 76311403 Ki = 3700 nM T13201 C5RAC6 76311404 Ki = 39 nM T13201 CY0R8X 76311405 Ki = 400 nM T13201 C7SO0T 76311406 Ki = 970 nM T13201 CYQ7B0 76311407 Ki = 950 nM T13201 CDGN83 76311408 Ki = 40 nM T13201 C4S6CE 76311409 Ki = 31 nM T13201 CTJ63S 76311410 Ki = 30 nM T13201 CEW21K 76311421 Ki = 650 nM T13201 C96NRT 76311425 Ki = 910 nM T13201 CG2JI0 76313836 Ki = 1568 nM T13201 CD1A5Y 76313837 Ki = 985 nM T13201 CU48XE 76313838 Ki = 4230 nM T13201 C04EFJ 76313840 Ki = 5328 nM T13201 CZ60NF 76313841 Ki = 6506 nM T13201 C5S3XY 76313842 Ki = 6428 nM T13201 CK2LR8 76313848 Ki = 274 nM T13201 CI3WQ5 76313849 Ki = 198 nM T13201 CB2YP3 76313998 Ki = 28000 nM T13201 C0KVD7 76314143 Ki > 10000 nM T13201 CE1H8W 76314144 Ki > 10000 nM T13201 C5EM0L 76314145 Ki > 10000 nM T13201 C0T8HW 76314452 Ki > 10000 nM T13201 CZ0JC7 76314453 Ki = 166 nM T13201 CC1Z6A 76314549 Ki > 50000 nM T13201 CA1F9S 76314550 Ki > 50000 nM T13201 CZBG52 76314647 Ki = 39 nM T13201 C4F7WP 76314648 Ki = 179 nM T13201 C95DKS 76314709 Ki > 10000 nM T13201 C37XBL 76314710 Ki > 10000 nM T13201 C2H7ZA 76314711 Ki > 10000 nM T13201 CE1BX4 76314958 Ki = 9200 nM T13201 C9R2KH 76314959 Ki = 4000 nM T13201 C1S9BI 76314960 Ki = 22 nM T13201 CRO70P 76314961 Ki = 56 nM T13201 C06NML 76314962 Ki = 617 nM T13201 C81HKS 76314963 Ki = 12000 nM T13201 CY9J1C 76314964 Ki = 500 nM T13201 C9W7DT 76314988 Ki = 35 nM T13201 C5JFN2 76314989 Ki = 1230 nM T13201 CKRF91 76314990 Ki = 67 nM T13201 C3C4PI 76315011 Ki = 9500 nM T13201 C20MYC 76315012 Ki = 3300 nM T13201 C34MRW 76317361 Ki = 843 nM T13201 CXZU92 76317371 Ki = 2456 nM T13201 CL5CF8 76317538 Ki > 100000 nM T13201 CB1VD3 76317966 Ki = 410 nM T13201 C6GOE1 76318042 Ki = 170 nM T13201 CGQ67N 76318218 Ki = 36 nM T13201 CLC1H8 76318279 Ki > 10000 nM T13201 CT7G2Z 76318280 Ki > 10000 nM T13201 CCO80M 76318281 Ki > 10000 nM T13201 CY5O9B 76318282 Ki > 10000 nM T13201 CM5IV7 76318283 Ki > 10000 nM T13201 C4DMY8 76318284 Ki > 10000 nM T13201 CG8QV5 76318285 Ki > 10000 nM T13201 CO18PL 76318590 Ki = 360 nM T13201 C98SVG 76318591 Ki = 120 nM T13201 CH14IG 76318592 Ki = 41 nM T13201 CYXT21 76318593 Ki = 250 nM T13201 C4J9XP 76318594 Ki = 71 nM T13201 CW59AZ 76318595 Ki = 77 nM T13201 COY1X4 76318596 Ki = 30 nM T13201 CU3R6B 76318626 Ki = 21300 nM T13201 CT94VN 76318627 Ki = 7050 nM T13201 CX2D4V 76318628 Ki = 700 nM T13201 C8SZQ7 76318648 Ki = 550 nM T13201 CFX3A2 76318651 Ki = 514 nM T13201 C1DC8O 76318659 Ki = 410 nM T13201 CDGH94 76321081 Ki = 529 nM T13201 CQ5B4S 76321082 Ki = 4560 nM T13201 C9U3LR 76321089 Ki = 4519 nM T13201 CZ2RY8 76321096 Ki = 341 nM T13201 CJM27E 76321273 Ki = 598 nM T13201 C9AP8I 76321274 Ki = 64000 nM T13201 C82NGW 76321408 Ki > 10000 nM T13201 CWM9C3 76321409 Ki = 501 nM T13201 C78KRT 76321425 Ki > 10000 nM T13201 CJ20ZB 76321688 Ki = 4350 nM T13201 CVT3O8 76321689 Ki = 1375 nM T13201 CH36SX 76321755 Ki = 868 nM T13201 C8SZN7 76321756 Ki = 8450 nM T13201 CP24WC 76321814 Ki > 10000 nM T13201 CNP1B7 76321907 Ki = 9.6 nM T13201 C4YP7A 76321908 Ki = 91 nM T13201 CZ31AU 76322240 Ki = 20000 nM T13201 C0GF7P 76322242 Ki = 1100 nM T13201 CQ5Z3H 76322243 Ki = 1050 nM T13201 CIS24L 76322244 Ki = 1500 nM T13201 CJN27S 76322270 Ki = 1280 nM T13201 C63TZU 76322272 Ki = 3780 nM T13201 C4T0DK 76322273 Ki = 625 nM T13201 CYZO10 76322274 Ki = 37 nM T13201 C1KL6D 76322275 Ki = 48 nM T13201 C7QUH8 76322276 Ki = 61 nM T13201 C1YDG3 76322277 Ki = 66 nM T13201 CG37HT 76322303 Ki = 27500 nM T13201 CZ98LC 76324732 Ki = 341 nM T13201 CW87DO 76324733 Ki = 4329 nM T13201 C5JXE8 76324738 Ki = 5867 nM T13201 CUG2O8 76324739 Ki = 5329 nM T13201 CLN0I8 76325020 Ki > 10000 nM T13201 C35EUT 76325021 Ki > 10000 nM T13201 CZQ93S 76325300 Ki = 447 nM T13201 CP3X6L 76325374 Ki = 220 nM T13201 CO79TZ 76325375 Ki = 711 nM T13201 CE1DM0 76325376 Ki = 292 nM T13201 CE3P4W 76325377 Ki > 10000 nM T13201 C7ZJ9M 76325378 Ki = 86 nM T13201 CN6CY7 76325452 Ki > 50000 nM T13201 CUC3M2 76325547 Ki = 12.1 nM T13201 C1BC4A 76325548 Ki = 7.9 nM T13201 CQUE95 76325602 Ki > 10000 nM T13201 CDO73V 76325603 Ki > 10000 nM T13201 C95MSJ 76325864 Ki = 21400 nM T13201 C73WKZ 76325865 Ki = 420 nM T13201 CB28DH 76325866 Ki = 295 nM T13201 CV0TP6 76325867 Ki = 521 nM T13201 C68YJL 76325868 Ki = 59 nM T13201 CMRD93 76325869 Ki = 39 nM T13201 C98JBS 76325870 Ki = 25500 nM T13201 CE5N1J 76325871 Ki = 190 nM T13201 CL0XR7 76325899 Ki = 48 nM T13201 CLI14U 76325900 Ki = 720 nM T13201 C7FI3X 76325901 Ki = 350 nM T13201 C27YJP 76325902 Ki = 780 nM T13201 C4KG1E 76325903 Ki = 21000 nM T13201 C4T0VX 76325904 Ki = 8100 nM T13201 CO14TP 76325929 Ki = 32 nM T13201 C9F1ZI 76325930 Ki = 39 nM T13201 CWP61T 76325931 Ki = 268 nM T13201 C0UK2H 76328279 Ki = 674 nM T13201 CCNB68 76328280 Ki = 4451 nM T13201 C8AS9R 76328281 Ki = 3781 nM T13201 C3D2QL 76328449 Ki = 133 nM T13201 CI47ZC 76328450 Ki = 3240 nM T13201 CM05DY 76328451 Ki = 47000 nM T13201 CN0KZ1 76328452 Ki = 47600 nM T13201 C0CFZ1 76328574 Ki = 490 nM T13201 CYM2G9 76328575 Ki = 522 nM T13201 CZ5X4W 76328576 Ki = 295 nM T13201 CP3CN4 76328593 Ki > 10000 nM T13201 CPJM79 76328853 Ki = 2365 nM T13201 C6F4LU 76328915 Ki = 507 nM T13201 C5VW9J 76328916 Ki > 10000 nM T13201 CEZ6A8 76328917 Ki = 6630 nM T13201 CYD50A 76329098 Ki = 3.9 nM T13201 CB23PR 76329099 Ki = 21.5 nM T13201 C3QI6J 76329100 Ki = 257 nM T13201 CTF2G1 76329169 Ki > 10000 nM T13201 CAE23D 76329170 Ki > 10000 nM T13201 CX8Z5D 76329449 Ki = 225 nM T13201 CUHX10 76329450 Ki = 23000 nM T13201 CU42FB 76329451 Ki = 343 nM T13201 CC69YL 76329452 Ki = 1150 nM T13201 C0HJ4Y 76329453 Ki = 1000 nM T13201 C3MO2T 76329454 Ki = 450 nM T13201 CEG87T 76329456 Ki = 6300 nM T13201 C7WV9M 76329457 Ki = 45 nM T13201 CVWR30 76329482 Ki = 210 nM T13201 CK5S6A 76329483 Ki = 130 nM T13201 CQ85UG 76329484 Ki = 12750 nM T13201 CPB5U8 76329485 Ki = 47 nM T13201 C6P5UM 76329498 Ki = 20100 nM T13201 C6H4KZ 76329499 Ki = 3400 nM T13201 CKH0X7 76331969 Ki = 1240 nM T13201 CO82ZX 76331970 Ki = 1528 nM T13201 C5U7JI 76331976 Ki = 5489 nM T13201 CYC39A 76331984 Ki = 276 nM T13201 CK73VH 76331985 Ki = 761 nM T13201 C5HRL1 76332129 Ki = 516 nM T13201 C68DOK 76332270 Ki > 10000 nM T13201 CJN0W8 76332271 Ki > 10000 nM T13201 C3ZGF1 76332272 Ki > 10000 nM T13201 C6ENW5 76332521 Ki = 354 nM T13201 C4RPU5 76332522 Ki = 1070 nM T13201 C14UQS 76332523 Ki = 2540 nM T13201 CGLB34 76332602 Ki = 89 nM T13201 CP9SU7 76332603 Ki > 10000 nM T13201 CG3U6D 76332757 Ki = 32 nM T13201 CSN84K 76332758 Ki = 54 nM T13201 COZ89H 76332830 Ki > 10000 nM T13201 CFI5K7 76332831 Ki > 10000 nM T13201 C5VN9Q 76332832 Ki > 10000 nM T13201 CG9HO7 76333094 Ki = 210 nM T13201 CNB7Q0 76333095 Ki = 12000 nM T13201 CNJF36 76333096 Ki = 285 nM T13201 CN1JW9 76333097 Ki = 200 nM T13201 CXA5T0 76333098 Ki = 365 nM T13201 CG60RB 76333099 Ki = 200 nM T13201 CJZM43 76333100 Ki = 600 nM T13201 C3K8WP 76333101 Ki = 36 nM T13201 CQRM32 76333124 Ki = 3450 nM T13201 CDY7R8 76333125 Ki = 7440 nM T13201 C8MYW5 76333126 Ki = 32100 nM T13201 CEP14I 76333127 Ki = 98 nM T13201 C9H4OK 76333128 Ki = 415 nM T13201 CH0YG6 76333129 Ki = 200 nM T13201 C98APF 76333130 Ki = 200 nM T13201 CNH71G 76333131 Ki = 415 nM T13201 C3NQY6 76333149 Ki = 1200 nM T13201 CVS5Z9 76333154 Ki = 22100 nM T13201 C9W0HZ 76335546 Ki = 2387 nM T13201 CZC97G 76335551 Ki = 3478 nM T13201 CK5I4M 76335747 Ki = 72200 nM T13201 CQKW51 76335889 Ki > 10000 nM T13201 CB53XC 76335911 Ki > 10000 nM T13201 CP16NU 76336199 Ki = 84 nM T13201 C3P4ZB 76336200 Ki = 132 nM T13201 CLB17E 76336381 Ki = 9.6 nM T13201 CV1B6C 76336382 Ki = 39.8 nM T13201 CWFY73 76336452 Ki > 10000 nM T13201 C2QC4D 76336453 Ki > 10000 nM T13201 CF1PD0 76336721 Ki = 885 nM T13201 CS7E0I 76336722 Ki = 600 nM T13201 C5RLH3 76336723 Ki = 62 nM T13201 CXM1A2 76336724 Ki = 8400 nM T13201 CO29MN 76336726 Ki = 200 nM T13201 CZ78TW 76336727 Ki = 15000 nM T13201 CT9V4M 76336730 Ki = 44 nM T13201 C0VCW9 76336761 Ki = 30 nM T13201 CO21QC 76336762 Ki = 120 nM T13201 C4JB8L 76336763 Ki = 800 nM T13201 CAN2Y3 76336778 Ki = 91 nM T13201 CM67SN 76336780 Ki = 890 nM T13201 CMV08B 76336782 Ki = 300 nM T13201 C5SEZ2 76336785 Ki = 180 nM T13201 CH0OY6 78319159 Ki > 50000 nM T13201 CC4F0A 78319160 Ki > 50000 nM T13201 CO4IE9 78319161 Ki > 50000 nM T13201 CY6LN4 78319162 Ki = 270 nM T13201 CU9I6V 82078731 Ki = 546.7 nM T13201 C5TB6O 82080973 Ki = 1274 nM T13201 CX5WB9 82198349 Ki = 765 nM T13201 C6UZR9 82911195 Ki = 2340 nM T13201 CVD64Q 83379931 Ki > 10000 nM T13201 CR47YB 86047482 Ki = 563 nM T13201 C0P3OF 86047486 Ki = 620 nM T13201 CZ5HA6 86047495 Ki = 667 nM T13201 CTD2Y9 86276273 Ki = 572 nM T13201 CHY2O4 86276274 Ki = 498 nM T13201 CN7HU3 86288843 Ki > 50000 nM T13201 C5Y1WO 86288855 Ki > 50000 nM T13201 C76RBA 86298624 IC50 = 6170 nM T13201 C93FKI 86298625 IC50 = 41 nM T13201 CVLU48 86298626 IC50 = 9030 nM T13201 CR97VD 86692717 Ki = 41.2 nM T13201 C8PC3U 86692718 Ki = 6.1 nM T13201 C6HC8V 86692720 Ki = 4014 nM T13201 CQ30FJ 86719933 Ki > 200000 nM T13201 CH2X9D 88314331 Ki > 10000 nM T13201 C3EYT4 88314336 Ki > 10000 nM T13201 CB4KI9 88973647 Ki = 532 nM T13201 C1O5YX 90180909 Ki > 200000 nM T13201 CIJ96H 90644155 IC50 > 10000 nM T13201 CX7EW1 90644156 IC50 > 10000 nM T13201 CK5GZ4 90644157 IC50 > 10000 nM T13201 C7O1YN 90644158 IC50 > 10000 nM T13201 CEN6C1 90644159 IC50 > 10000 nM T13201 C8X9UZ 90644160 IC50 > 10000 nM T13201 C6I9RG 90644374 Ki = 3930 nM T13201 C1DT9W 90644375 Ki = 4010 nM T13201 C2PXK3 90644376 Ki = 3660 nM T13201 C7OJM0 90644377 Ki = 3620 nM T13201 C3Z8QO 90644378 Ki = 2880 nM T13201 C4QT6W 90644479 Ki = 573 nM T13201 C6XB9R 90644480 Ki = 1165 nM T13201 C1KXA0 90644481 Ki = 934 nM T13201 C1ND2E 90644482 Ki = 1260 nM T13201 CY4LZ9 90644483 Ki = 5430 nM T13201 C2RQD9 90644484 Ki = 6400 nM T13201 CZ0R6T 90644485 Ki = 7355 nM T13201 C4G1BD 90644486 Ki = 6230 nM T13201 CL7I9M 90644487 Ki = 5490 nM T13201 CVMU79 90644488 Ki = 7200 nM T13201 C6F5ZP 90644489 Ki = 3470 nM T13201 CG85NB 90644490 Ki = 2750 nM T13201 CCID31 90644491 Ki = 3025 nM T13201 C3BPF8 90644492 Ki = 2400 nM T13201 C7B5YR 90644493 Ki = 643 nM T13201 C9FCX5 90644494 Ki = 718 nM T13201 CQND72 90644495 Ki = 1350 nM T13201 C4V9IZ 90644496 Ki = 1175 nM T13201 C49VLZ 90644497 Ki = 3200 nM T13201 CX2I9G 90644498 Ki = 2340 nM T13201 C5MXJ4 90644499 Ki = 568 nM T13201 C2E7QM 90644500 Ki = 671 nM T13201 CR02MV 90644501 Ki = 349 nM T13201 C2SZ5P 90644502 Ki = 1320 nM T13201 C86NMC 90644503 Ki = 2340 nM T13201 C8W3PI 90644504 Ki = 3200 nM T13201 CF12MK 90645415 Ki = 84.7 nM T13201 CJO6I7 90645416 Ki = 159.6 nM T13201 CU2K5R 90645417 Ki = 21.6 nM T13201 C58KIU 90645418 Ki = 32.4 nM T13201 CS0OX7 90645419 Ki = 66 nM T13201 CWD6P7 90645420 Ki = 27.6 nM T13201 CVY5P9 90645421 Ki = 33.2 nM T13201 CAL9C4 90645422 Ki = 23.2 nM T13201 C2EA9C 90645423 Ki = 28.4 nM T13201 C1FVA8 90645424 Ki = 94.1 nM T13201 CP27AX 90645425 Ki = 69.1 nM T13201 C8E4ZH 90645426 Ki = 25.4 nM T13201 C3SIA9 90645429 Ki = 498 nM T13201 C1E4FS 90645430 Ki = 25.1 nM T13201 COBQ09 90645431 Ki = 16.3 nM T13201 C7IU8K 90645432 Ki = 28.2 nM T13201 CW0L1D 90654798 Ki > 50000 nM T13201 CO2CU1 90654800 Ki > 50000 nM T13201 CE54MK 90654802 Ki > 50000 nM T13201 CID9U2 90654804 Ki > 50000 nM T13201 C27QHW 90654822 Ki = 4930 nM T13201 C96OWE 90654823 Ki > 50000 nM T13201 CZQ9E3 90654824 Ki > 50000 nM T13201 CCPO43 90654825 Ki = 8025 nM T13201 C4D2TM 90654826 Ki = 5320 nM T13201 C48XBN 90654827 Ki > 50000 nM T13201 CI8TG3 90654828 Ki = 8745 nM T13201 C6GFZ0 90654829 Ki = 354 nM T13201 C3Z1GS 90654830 Ki > 50000 nM T13201 C4JSW5 90655322 Ki = 497 nM T13201 C3QH0R 90655323 Ki = 521 nM T13201 CF0U7K 90655324 Ki = 411 nM T13201 C3OL7F 90656456 Ki = 30.3 nM T13201 CM10BY 90656457 Ki = 25.5 nM T13201 CGOV47 90656459 Ki = 76 nM T13201 CM3HC6 90656461 Ki = 59.5 nM T13201 CA9L3I 90656462 Ki = 51.9 nM T13201 C6F0AY 90656464 Ki = 665 nM T13201 CE0F5O 90656465 Ki = 50.3 nM T13201 CX4I7B 90656468 Ki = 56.05 nM T13201 CZ80KF 90656469 Ki = 251.5 nM T13201 CX4YM5 90656470 Ki = 18.75 nM T13201 CU31VY 90675933 Ki > 10000 nM T13201 C2XWG7 90675934 Ki > 10000 nM T13201 CH7R2B 90675935 Ki > 10000 nM T13201 CORQ94 90675936 Ki > 10000 nM T13201 CE39DC 90675937 Ki > 10000 nM T13201 CSU5K2 90675938 Ki > 10000 nM T13201 CE8S1J 90675939 Ki > 10000 nM T13201 C1H9FB 90675940 Ki > 10000 nM T13201 CPB36R 90675941 Ki > 10000 nM T13201 C3SJ1D 90677341 Ki = 93 nM T13201 CK1GA3 90677342 Ki = 72 nM T13201 C0CR6D 90681501 Ki = 6780 nM T13201 C28FLQ 91498333 Ki > 10000 nM T13201 CE6LO5 91595667 Ki = 96.3 nM T13201 C3AYZ5 91811067 Ki = 5783 nM T13201 CQF98O 91827503 Ki = 78.6 nM T13201 C3I6NV 91827505 Ki = 76.2 nM T13201 CW1P4E 91827506 Ki = 8.5 nM T13201 CE2OY1 91995964 Ki = 62 nM T13201 CX45AP 92044053 Ki = 2560 nM T13201 CEH68Q 93972064 Ki = 149.5 nM T13201 C28QRZ 101564149 Ki = 79100 nM T13201 CE8GH2 101874826 Ki = 21.6 nM T13201 C4W9FG 101874827 Ki = 64.2 nM T13201 CY7G8A 101874828 Ki = 52.8 nM T13201 C1TM8I 101874829 Ki = 57.8 nM T13201 CVZ3L5 101874830 Ki = 82.6 nM T13201 C2H5FC 101876957 Ki = 215 nM T13201 CDGZ03 101879106 Ki = 32.2 nM T13201 CY6ER7 101879108 Ki = 41.8 nM T13201 C04YZS 101913644 Ki = 803 nM T13201 CAC1W7 101913750 Ki = 6650 nM T13201 CQX8K1 101913751 Ki = 7440 nM T13201 CIP25Q 101913752 Ki = 8690 nM T13201 CTY15S 101913753 Ki > 50000 nM T13201 C49NEJ 101913754 Ki = 7210 nM T13201 CW5Q7L 101913755 Ki = 8670 nM T13201 CE90SD 102138248 Ki = 347 nM T13201 CB1PK8 102151146 Ki = 23200 nM T13201 C0A6FY 102151151 Ki > 100000 nM T13201 CP1X9Y 102232756 Ki = 690 nM T13201 C1XV9H 102311866 Ki = 67300 nM T13201 CQBE51 102341119 Ki = 9500 nM T13201 C2TX7A 102354117 Ki = 1335 nM T13201 CK43QR 102405972 Ki = 8360 nM T13201 C0CVO4 102480165 Ki = 52100 nM T13201 C6LUE5 109059506 Ki = 307 nM T13201 CUY64D 109061586 Ki > 10000 nM T13201 C20JDY 110347401 Ki = 100400 nM T13201 CXN7Z8 110453853 Ki = 2397 nM T13201 C6I0LD 112499923 Ki = 2340 nM T13201 C8CFR6 112499924 Ki = 146 nM T13201 C74UZL 112684088 Ki = 0.2747 nM T13201 CK52CI 112686058 Ki = 0.6571 nM T13201 CP5B7N 112687648 Ki = 0.4794 nM T13201 CUR4V8 114816322 Ki > 10000 nM T13201 C3TZ9A 115950959 Ki = 24.8 nM T13201 CAO67C 118705769 Ki = 15.9 nM T13201 CW1D8A 118705770 Ki = 12.4 nM T13201 CTFB51 118705771 Ki = 8.5 nM T13201 C5NGT8 118705772 Ki = 16 nM T13201 C3G4ZN 118705773 Ki = 19.8 nM T13201 CBVD13 118705774 Ki = 21.1 nM T13201 C3KCZ6 118705775 Ki = 492 nM T13201 C5Z4QF 118705776 Ki = 591 nM T13201 CV4YN0 118705777 Ki = 214 nM T13201 C0IBQ8 118705778 Ki = 498 nM T13201 CH7LV5 118705779 Ki = 244 nM T13201 CU5SI9 118705780 Ki = 262 nM T13201 C6IGP0 118705781 Ki = 303 nM T13201 C7ZE2H 118705782 Ki = 282 nM T13201 C47QFN 118705783 Ki = 387 nM T13201 CO1P3T 118705784 Ki = 354 nM T13201 CK8E5C 118705785 Ki = 337 nM T13201 CS9G2U 118705786 Ki = 229 nM T13201 C1XV9M 118705787 Ki = 101 nM T13201 C7GW3Q 118705788 Ki = 106 nM T13201 CUIS94 118706141 Ki = 9.5 nM T13201 CET19U 118706142 Ki = 103 nM T13201 C6FBG3 118706893 Ki = 319 nM T13201 C1CLV5 118706959 Ki = 346 nM T13201 CLA5I2 118706960 Ki = 344 nM T13201 C8GD4Y 118706961 Ki = 327 nM T13201 CB0E4N 118706962 Ki = 354 nM T13201 CFX37I 118707439 Ki = 19.8 nM T13201 CURF40 118707440 Ki = 253 nM T13201 C2SPI1 118707441 Ki = 2270 nM T13201 CK7VG2 118707442 Ki = 517 nM T13201 CB6IF2 118707443 Ki = 193 nM T13201 C5O1TK 118707444 Ki = 267 nM T13201 C5VW3Z 118707445 Ki = 972 nM T13201 CM5Z7B 118707446 Ki = 2120 nM T13201 CANH39 118707447 Ki = 484 nM T13201 CQO91H 118707448 Ki = 430 nM T13201 C2PU1D 118707449 Ki = 2330 nM T13201 C8H7SM 118707452 Ki = 626 nM T13201 CYJ0I7 118707453 Ki = 2310 nM T13201 C0R9FG 118707454 Ki = 519 nM T13201 CJI04D 118707455 Ki = 3150 nM T13201 CO8AF6 118707456 Ki = 289 nM T13201 CJP1W6 118707457 Ki = 6030 nM T13201 C3G0AY 118707458 Ki = 22.1 nM T13201 CM1B4X 118707459 Ki = 151.3 nM T13201 C0WO2M 118707460 Ki = 88.9 nM T13201 CKV43U 118710106 Ki = 2343 nM T13201 CBAQ59 118710108 Ki = 960.5 nM T13201 CPI7L3 118710135 Ki > 20000 nM T13201 C05ZCN 118710136 Ki > 20000 nM T13201 C45XHE 118710137 Ki > 20000 nM T13201 C84YKV 118710138 Ki = 2900 nM T13201 CFA76H 118710139 Ki = 15650 nM T13201 C0UWK2 118710140 Ki = 2485 nM T13201 CGJ59E 118710141 Ki > 20000 nM T13201 C64BUR 118710142 Ki > 20000 nM T13201 C1W2DB 118710143 Ki > 20000 nM T13201 CZ4F3O 118710144 Ki > 20000 nM T13201 CWR82N 118710145 Ki > 20000 nM T13201 C7R5FO 118710146 Ki > 20000 nM T13201 CD8U1O 118710147 Ki > 20000 nM T13201 C8YFH6 118710148 Ki > 20000 nM T13201 CLPC68 118710149 Ki > 20000 nM T13201 C8OH4V 118710150 Ki > 20000 nM T13201 C6CAQ4 118710151 Ki > 20000 nM T13201 CS0G7T 118710152 Ki > 20000 nM T13201 C3NPF1 118710200 Ki > 20000 nM T13201 C4YXF1 118710201 Ki > 20000 nM T13201 C1B5QL 118710202 Ki > 20000 nM T13201 CUJ42P 118710203 Ki = 1300 nM T13201 CK23DF 118710598 Ki = 41.2 nM T13201 CS9MC2 118710599 Ki = 82.3 nM T13201 CW2D4O 118710600 Ki = 40.2 nM T13201 CTMF04 118710601 Ki = 48.9 nM T13201 CU2C9L 118710602 Ki = 47.7 nM T13201 CFCG50 118710603 Ki = 49.3 nM T13201 C2G5DI 118710604 Ki = 52.5 nM T13201 CY2S9V 118710605 Ki = 47 nM T13201 C5L6IK 118710606 Ki = 41.3 nM T13201 C6ZGB2 118711612 Ki = 357 nM T13201 CNS6L8 118711613 Ki = 3200 nM T13201 CY0E8G 118711614 Ki = 1250 nM T13201 CI71PW 118711615 Ki = 1185 nM T13201 C1X7RI 118711616 Ki = 1350 nM T13201 C7P6GM 118711617 Ki = 1500 nM T13201 CYNA84 118711618 Ki = 413 nM T13201 CL38UN 118711619 Ki = 42.1 nM T13201 CGUV98 118711620 Ki = 41.5 nM T13201 CJ2UH6 118711621 Ki = 1450 nM T13201 CH2RE7 118711622 Ki = 416 nM T13201 C1RWN4 118711623 Ki = 652 nM T13201 CR0I6S 118711624 Ki = 835 nM T13201 C8LQI3 118711625 Ki = 258 nM T13201 C5SEJ6 118711626 Ki = 44.9 nM T13201 C5TYE7 118711627 Ki = 330 nM T13201 C7ZOH6 118712658 Ki = 5670 nM T13201 C19IXJ 118712659 Ki > 50000 nM T13201 CD5MB4 118712660 Ki = 4670 nM T13201 C0EPI8 118712661 Ki = 7480 nM T13201 CUO2I5 118714986 Ki = 105 nM T13201 CHL5P7 118714987 Ki = 119 nM T13201 CKGY64 118714988 Ki = 86.5 nM T13201 CQ3L5G 118714989 Ki = 2078 nM T13201 CK9FR8 118714990 Ki = 4761 nM T13201 CVM9K5 118714991 Ki = 5432 nM T13201 CXP7N8 118714992 Ki = 674 nM T13201 C0OE2J 118714993 Ki = 3371 nM T13201 CN26WF 118715053 Ki = 4168 nM T13201 C6RIG2 118715054 Ki = 793 nM T13201 C9T4CK 118715055 Ki = 2162 nM T13201 C19IQV 118715056 Ki = 4549 nM T13201 CZ18GD 118716360 Ki = 1050 nM T13201 CX6F4B 118716361 Ki = 1350 nM T13201 CO4K8Z 118716362 Ki = 350 nM T13201 CR8HX4 118716363 Ki = 2400 nM T13201 CYH2P1 118716364 Ki = 1550 nM T13201 C61BOY 118716365 Ki > 20000 nM T13201 C8PJC3 118716366 Ki = 9000 nM T13201 C9HP7J 118716367 Ki = 2400 nM T13201 CTS52R 118716368 Ki > 20000 nM T13201 CHI60Z 118716369 Ki = 2400 nM T13201 CA1UY4 118716496 Ki = 198 nM T13201 CVR32C 118716497 Ki = 377 nM T13201 CT1RQ6 118716498 Ki = 479 nM T13201 CG10AC 118716499 Ki = 414 nM T13201 CV89MK 118716500 Ki = 483 nM T13201 C57YMW 118716501 Ki = 887 nM T13201 CQ73KL 118716502 Ki = 283 nM T13201 CXE59K 118716504 Ki = 1870 nM T13201 CONM87 118716505 Ki = 704 nM T13201 CQ3I7N 118716509 Ki = 40.7 nM T13201 C72KER 118716510 Ki = 214 nM T13201 C0RJI1 118716511 Ki = 147 nM T13201 CFU0Z8 118716512 Ki = 218 nM T13201 CXU4D7 118716513 Ki > 10000 nM T13201 C86KQZ 118716514 Ki > 10000 nM T13201 C9HLA8 118716891 Ki = 813 nM T13201 CJ0YC9 118716892 Ki = 752 nM T13201 CJ8TZ3 118716893 Ki > 10000 nM T13201 C0X1WQ 118716894 Ki > 10000 nM T13201 CDG4L8 118716895 Ki > 10000 nM T13201 CFD26B 118716950 Ki = 4372 nM T13201 C20YBM 118716951 Ki = 3055 nM T13201 C0V1ZT 118716952 Ki = 499 nM T13201 CH9BW0 118716953 Ki = 248 nM T13201 CXB89Y 118716954 Ki = 1511 nM T13201 C8CKU2 118716955 Ki = 7005 nM T13201 CYN29C 118716960 Ki = 1345 nM T13201 C4AC7H 118716961 Ki = 2940 nM T13201 CJ9O3I 118716962 Ki = 2190 nM T13201 C6RJ9W 118716964 Ki = 2630 nM T13201 CMVW90 118716999 Ki > 10000 nM T13201 CBKN39 118717000 Ki = 917 nM T13201 C6N8CF 118717001 Ki = 927 nM T13201 CL3P7I 118717002 Ki > 10000 nM T13201 C2H0NP 118717003 Ki > 10000 nM T13201 CXRD23 118719969 Ki = 72.8 nM T13201 C4Z6DI 118719970 Ki = 57.6 nM T13201 C2HJ4Y 118719971 Ki > 10000 nM T13201 CD1OH8 118719972 Ki > 10000 nM T13201 C0R8JN 118719973 Ki = 4970 nM T13201 CMR0H2 118719974 Ki = 5735 nM T13201 CI3QG5 118719975 Ki > 10000 nM T13201 C06YTV 118719976 Ki = 2380 nM T13201 C25BJT 118721385 Ki = 8806 nM T13201 CI4W0E 118721386 Ki = 7408 nM T13201 CFRX59 118721387 Ki = 10316 nM T13201 C5SYD7 118721388 Ki = 15690 nM T13201 CNT18B 118721389 Ki = 2630 nM T13201 CYC50E 118721390 Ki = 2331 nM T13201 CYL0W1 118721391 Ki = 157 nM T13201 C1HN6R 118721392 Ki = 268 nM T13201 C2WLI4 118721393 Ki = 690 nM T13201 CQVS30 118721394 Ki = 313 nM T13201 CL2Q8M 118721395 Ki = 407 nM T13201 CAG5L6 118721396 Ki = 381 nM T13201 CJ63BR 118721397 Ki = 9818 nM T13201 C14ZNT 118721398 Ki > 50000 nM T13201 C1J6IX 118721399 Ki > 50000 nM T13201 CVJ92D 118721400 Ki = 12108 nM T13201 C5F7PT 118721401 Ki > 50000 nM T13201 C5AFR3 118721402 Ki > 50000 nM T13201 C29EYL 118721403 Ki = 28679 nM T13201 C8GYO9 118721404 Ki = 29070 nM T13201 CSZ7Q0 118721405 Ki > 50000 nM T13201 CY3ZW6 118721406 Ki = 7161 nM T13201 C4T9IR 118721407 Ki = 26810 nM T13201 CNPB81 118721408 Ki = 23102 nM T13201 CP40JF 118722001 Ki > 10000 nM T13201 CXTR97 118723294 Ki = 5.3 nM T13201 C42JBV 118723295 Ki = 6.6 nM T13201 CVDC56 118723296 Ki = 7.9 nM T13201 C2RG7F 118723303 Ki = 18 nM T13201 C0CMO4 118723304 Ki = 17.1 nM T13201 CC7RH0 118723305 Ki = 90.9 nM T13201 CU0R8X 118723306 Ki = 826 nM T13201 C67LPC 118723308 Ki = 151 nM T13201 C0D1SQ 118724328 Ki = 373.4 nM T13201 C89YTC 118724329 Ki = 359 nM T13201 CBT87C 118724330 Ki = 214.4 nM T13201 C49AWZ 118724331 Ki = 52.6 nM T13201 CP9X5K 118728047 Ki = 85.9 nM T13201 CUA3S7 118728048 Ki = 706 nM T13201 C2K3DO 118728049 Ki = 295 nM T13201 CZTN86 118728050 Ki = 66.5 nM T13201 C0CUV2 118728051 Ki = 494 nM T13201 CGU5O0 118728053 Ki = 240 nM T13201 CGQ69F 118728055 Ki = 615 nM T13201 C2JEW0 118728057 Ki = 485 nM T13201 CCBJ19 118728058 Ki = 290 nM T13201 CKJ8S9 118728060 Ki = 496 nM T13201 C0O3BI 118728062 Ki = 109 nM T13201 CH2E8F 118728064 Ki = 910 nM T13201 C4JM1O 118728066 Ki = 683 nM T13201 C67YPT 118728068 Ki = 434 nM T13201 CML9F8 118728070 Ki = 84.7 nM T13201 CA52IR 118728072 Ki = 415 nM T13201 CVE9H5 118728074 Ki = 97.5 nM T13201 CS9ZW3 118728500 Ki > 10000 nM T13201 CI7MY8 118728501 Ki > 10000 nM T13201 CZE9K8 118728502 Ki > 10000 nM T13201 C8S9JV 118728503 Ki = 6831 nM T13201 COJB53 118728998 IC50 = 178.7 nM T13201 C4GJ2A 118728999 IC50 = 132.9 nM T13201 C16CPW 118729000 IC50 = 153.1 nM T13201 CRH8X5 118729001 Ki = 122.8 nM T13201 CD97RL 118729002 Ki = 36.4 nM T13201 C19HNU 118729003 Ki = 97.3 nM T13201 C8IJ7W 118729004 IC50 = 210.2 nM T13201 CZLP09 118729005 Ki = 144.7 nM T13201 C1W9DT 118729006 Ki = 105.4 nM T13201 CS30QV 118729007 Ki = 51.7 nM T13201 C40AIB 118729374 Ki > 10000 nM T13201 CO3Z5E 118729375 Ki > 10000 nM T13201 C6S0DR 118729376 Ki > 10000 nM T13201 CVXO79 118729377 Ki > 10000 nM T13201 C62BGK 118729378 Ki > 10000 nM T13201 C4D9EP 118729379 Ki > 10000 nM T13201 C2TOH7 118729380 Ki > 10000 nM T13201 C5P9ND 118729381 Ki > 10000 nM T13201 C2XLV4 118729382 Ki > 10000 nM T13201 CVLK60 118729383 Ki > 10000 nM T13201 C8U7SE 118729384 Ki > 10000 nM T13201 CV7OS1 118729385 Ki > 10000 nM T13201 C7Z2OR 118729386 Ki > 10000 nM T13201 CHE1K4 118729473 Ki = 231 nM T13201 C9V8MA 118729474 Ki = 3450 nM T13201 C8GJP5 118729475 Ki = 5675 nM T13201 C4MEZ0 118729476 Ki = 2418 nM T13201 CE3IV5 118729477 Ki = 6400 nM T13201 C5DM9L 118731312 Ki = 3 nM T13201 C7EX8M 118732578 Ki = 7445 nM T13201 C0A2SM 118732579 Ki = 20000 nM T13201 CV2JZ8 118732580 Ki = 3190 nM T13201 C2GNO4 118732581 Ki = 5665 nM T13201 CES83M 118732582 Ki = 141 nM T13201 CF2WQ4 118732583 Ki = 87 nM T13201 C08EZC 118733945 Ki > 10000 nM T13201 C3F1DU 118733947 Ki > 10000 nM T13201 C4OL1A 118733948 Ki > 10000 nM T13201 CP25HS 118733949 Ki > 10000 nM T13201 CY3H4E 118736318 Ki = 442 nM T13201 C8HY4S 118736320 Ki = 308 nM T13201 C7F5JH 118736322 Ki = 1696 nM T13201 C7MDJ3 118736324 Ki = 405 nM T13201 CQM67J 118736325 Ki = 7.2 nM T13201 CKY90W 118736326 Ki = 12.4 nM T13201 CY4B1U 118736327 Ki = 17 nM T13201 CRZ1T6 118736328 Ki = 44.9 nM T13201 CFDB97 118737265 Ki > 10000 nM T13201 CVGF86 118737267 Ki > 10000 nM T13201 C6B8WR 118737268 Ki > 10000 nM T13201 CWEM68 118737269 Ki > 10000 nM T13201 C6PXT8 118737270 Ki > 10000 nM T13201 CWP7Q1 118737271 Ki > 10000 nM T13201 CAB65M 118737272 Ki > 10000 nM T13201 CHR0I7 118737273 Ki > 10000 nM T13201 C72BLG 118737274 Ki > 10000 nM T13201 C4TD0Q 118737275 Ki > 10000 nM T13201 CZ1J0U 118737276 Ki > 10000 nM T13201 CHN09Y 118737277 Ki > 10000 nM T13201 CMR62B 118737278 Ki > 10000 nM T13201 C1CV3E 118737279 Ki > 10000 nM T13201 CUQ7H9 119082247 Ki = 1522.7 nM T13201 CP8Y5U 119090745 Ki > 10000 nM T13201 C4K6CG 119943184 Ki = 7120 nM T13201 CHX4Y2 121382833 Ki > 50000 nM T13201 CNEJ87 121382878 Ki = 73 nM T13201 CBHM75 121382881 Ki = 8400 nM T13201 C13GKC 121382882 Ki = 5580 nM T13201 C8QTR4 121382883 Ki = 5950 nM T13201 C96ANJ 121382897 Ki > 50000 nM T13201 CUS64J 121382999 Ki = 539 nM T13201 C6C4WE 121383002 Ki = 743 nM T13201 CG48HD 122164592 Ki = 6610 nM T13201 CK92MV 122179845 Ki = 467 nM T13201 C10UQY 122179846 Ki = 4490 nM T13201 CLV96C 122179847 Ki = 330 nM T13201 C2RT1Y 122179848 Ki = 605 nM T13201 C06ZSC 122179849 Ki = 810 nM T13201 C74RAE 122179850 Ki = 798 nM T13201 C6NM0Q 122179851 Ki = 3440 nM T13201 CYP3B0 122179852 Ki = 3715 nM T13201 CMP05I 122179853 Ki = 571 nM T13201 C2TGN6 122179854 Ki = 854 nM T13201 CAH3I1 122179855 Ki = 4215 nM T13201 CPKX90 122179856 Ki = 0.127 nM T13201 CQ2P5O 122179857 Ki = 0.1271 nM T13201 CVB9C4 122179858 Ki = 0.0483 nM T13201 CO6QP7 122179859 Ki = 0.1397 nM T13201 CP01MN 122179860 Ki = 0.0459 nM T13201 CJG71H 122179861 Ki = 0.6875 nM T13201 C8YJ9B 122180166 Ki > 10000 nM T13201 CHON20 122180167 Ki > 10000 nM T13201 C9L2TG 122180168 Ki > 10000 nM T13201 C9L3OY 122180169 Ki > 10000 nM T13201 CJ1X2F 122180170 Ki > 10000 nM T13201 CVCX92 122180171 Ki > 10000 nM T13201 C6LEA3 122180172 Ki > 10000 nM T13201 CV8Z4I 122182643 Ki = 182 nM T13201 CV96QP 122182644 Ki = 159 nM T13201 CA91HP 122182645 Ki = 222 nM T13201 C08EBQ 122182646 Ki = 258 nM T13201 CSJA24 122182647 Ki = 8.8 nM T13201 CDM51W 122182648 Ki = 27.1 nM T13201 C3E9FK 122182649 Ki = 26.5 nM T13201 CUF5N9 122182650 Ki = 49.4 nM T13201 C5BRH0 122182651 Ki = 54.1 nM T13201 C45DQE 122182654 Ki = 77.1 nM T13201 CDRF43 122182655 Ki = 160 nM T13201 CQ83BJ 122182656 Ki = 36.2 nM T13201 CH4Z8B 122182657 Ki = 12 nM T13201 CU71LK 122182658 Ki = 26.1 nM T13201 CY1NK4 122182659 Ki = 37.4 nM T13201 CP4I8D 122184891 Ki = 245 nM T13201 CZ2RM0 122184892 Ki = 32.5 nM T13201 CFQ4R3 122184893 Ki = 185 nM T13201 C69UQF 122184894 Ki = 143 nM T13201 CNF20A 122184895 Ki = 320 nM T13201 CJAL95 122184896 Ki = 20.7 nM T13201 C51LFX 122184933 Ki = 20.4 nM T13201 CTQP23 122184934 Ki = 26.7 nM T13201 CL49QM 122184935 Ki = 85.6 nM T13201 CVN28C 122184936 Ki = 1107 nM T13201 CU4S6Y 122184937 Ki = 23.3 nM T13201 C4VWG9 122184938 Ki = 149 nM T13201 C7H8ZI 122184984 Ki = 316.5 nM T13201 CX76HF 122184985 Ki = 896.8 nM T13201 C1KOF6 122184986 Ki = 9.4 nM T13201 C01CWK 122184987 Ki = 581.3 nM T13201 CVTY87 122184988 Ki = 851.5 nM T13201 CM5A7F 122184989 Ki = 63.5 nM T13201 CYM65N 122184990 Ki = 88.1 nM T13201 CQ9YU1 122184991 Ki = 282.4 nM T13201 C83GXC 122184992 Ki = 277.2 nM T13201 CTV40W 122184993 Ki = 290.9 nM T13201 CWM21G 122184994 Ki = 70.2 nM T13201 C19LDQ 122184995 Ki = 300.4 nM T13201 C7UE2C 122184996 Ki = 799.8 nM T13201 CWBN52 122184997 Ki > 10000 nM T13201 C1CI4W 122184998 Ki = 5296.1 nM T13201 CWJ94V 122185033 Ki = 350 nM T13201 C3G8EB 122185233 Ki = 464000 nM T13201 C9PG8Z 122185234 Ki > 10000 nM T13201 C93KBM 122185235 Ki = 1576 nM T13201 CX6Z5Y 122185236 Ki = 2108 nM T13201 CFPV38 122185237 Ki = 1767 nM T13201 CVZ70D 122185238 Ki = 1517 nM T13201 C14OHP 122185239 Ki = 2189 nM T13201 CB63WU 122185240 Ki = 838 nM T13201 CE3Q1J 122185241 Ki = 2167 nM T13201 CNG63S 122185242 Ki = 1925 nM T13201 CY7H0T 122185243 Ki = 1593 nM T13201 C2ME1I 122185244 Ki = 174 nM T13201 C0EPT7 122185245 Ki = 1.8 nM T13201 CI1AL4 122185246 Ki = 2226 nM T13201 CM43CE 122185684 Ki = 8039 nM T13201 CSQ43L 122185685 Ki = 7757 nM T13201 CCA9I1 122185686 Ki = 611 nM T13201 CLIR24 122185687 Ki = 128 nM T13201 C5NWU9 122185688 Ki = 1180 nM T13201 CY70TU 122185689 Ki = 652 nM T13201 CD94UC 122185690 Ki = 124 nM T13201 C8TIP4 122185692 Ki = 127 nM T13201 CE7W6O 122185694 Ki = 940 nM T13201 CV2G7S 122185695 Ki = 5924 nM T13201 C1M5JR 122185696 Ki = 304 nM T13201 CMB32C 122185697 Ki = 246 nM T13201 C1FR9Q 122185698 Ki = 230 nM T13201 CY2D9L 122185699 Ki = 264 nM T13201 C2NUJ9 122185700 Ki = 234 nM T13201 CHBC74 122185771 Ki = 271 nM T13201 CZM98F 122185772 Ki = 221 nM T13201 CP8Y5E 122185773 Ki = 215 nM T13201 CK2Q7M 122185774 Ki = 304 nM T13201 CF4L0N 122185776 Ki = 767 nM T13201 C7T4BF 122185778 Ki = 2740 nM T13201 C4TZ6G 122185779 Ki > 10000 nM T13201 CUI73A 122187162 Ki = 4.8 nM T13201 C1Q7AX 122187163 Ki = 55.3 nM T13201 CO6P7A 122187164 Ki = 0.01 nM T13201 C9LN8Q 122187165 Ki = 0.01 nM T13201 COK6D7 122187166 Ki = 45.4 nM T13201 C7NV8G 122187167 Ki = 289 nM T13201 C6XKH1 122187168 Ki = 231 nM T13201 C5KMW2 122187169 Ki > 10000 nM T13201 CSA78D 122187170 Ki > 10000 nM T13201 C5V7SZ 122187171 Ki = 6110 nM T13201 C6FMG1 122187172 Ki = 8.5 nM T13201 CVG1U0 122187173 Ki = 58.6 nM T13201 CR8NT0 122187174 Ki > 10000 nM T13201 CWSM36 122187175 Ki > 10000 nM T13201 CT59AR 122187176 Ki = 141 nM T13201 C93ESN 122187177 Ki = 130 nM T13201 CL0JF6 122187178 Ki = 36.8 nM T13201 CQ81UP 122187179 Ki = 41.9 nM T13201 CIE0W8 122187180 Ki = 22.5 nM T13201 CNSU27 122187181 Ki = 0.05 nM T13201 C7LDH1 122187182 Ki = 22 nM T13201 CG9T3N 122187183 Ki = 9 nM T13201 CBE9U8 122187184 Ki = 79.9 nM T13201 C13USE 122187185 Ki = 0.09 nM T13201 CE36PK 122187423 Ki = 213 nM T13201 CDS2I6 122187424 Ki = 1945 nM T13201 CMF63L 122187425 Ki > 10000 nM T13201 C7Q9TP 122187426 Ki = 9490 nM T13201 C04HSI 122187596 Ki = 31 nM T13201 CZ74KO 122187597 Ki = 300 nM T13201 C07OYV 122187598 Ki = 90 nM T13201 CO6AT2 122187599 Ki = 69 nM T13201 C7WJ4B 122187600 Ki = 37 nM T13201 CZ0Y1G 122187601 Ki = 55 nM T13201 CWF7Z0 122187602 Ki = 88 nM T13201 C07ZNW 122187603 Ki = 552 nM T13201 C7K6TV 122187604 Ki = 250 nM T13201 CX69YT 122187605 Ki = 50 nM T13201 C8XN0F 122187606 Ki = 64 nM T13201 CVT13C 122187607 Ki = 60 nM T13201 CB2DT8 122187638 Ki = 33.8 nM T13201 C0G4CQ 122187639 Ki = 931 nM T13201 CQSV13 122187640 Ki = 26.5 nM T13201 CH74EW 122187641 Ki = 51.6 nM T13201 CH3C8V 122187642 Ki = 7.5 nM T13201 CP01NQ 122187643 Ki = 43.8 nM T13201 CRM3S4 122188878 Ki = 437 nM T13201 C5UF1Q 122188879 Ki = 528 nM T13201 CQB9A8 122188880 Ki = 860 nM T13201 C1SFD4 122188881 Ki = 564 nM T13201 CIE7L0 122188882 Ki = 922 nM T13201 C6MPI4 122189078 Ki > 40000 nM T13201 C9V7WT 122189088 Ki > 40000 nM T13201 C1QZV7 122189098 Ki > 40000 nM T13201 CN16RY 122189300 Ki = 31 nM T13201 CYN3T8 122189301 Ki = 39.9 nM T13201 CSW9D1 122189302 Ki = 29 nM T13201 C6USQ7 122189303 Ki = 186 nM T13201 CQ4X1G 122189304 Ki = 58 nM T13201 C5XT3S 122192640 Ki = 5100 nM T13201 C1LCB9 122192641 Ki = 2500 nM T13201 CP51XT 122192642 Ki = 8870 nM T13201 C5GKT0 122192643 Ki = 2090 nM T13201 C3RZM8 122192644 Ki = 4550 nM T13201 CHLG86 122192645 Ki = 6920 nM T13201 CTK4J8 122192646 Ki = 6530 nM T13201 CVNQ49 122192647 Ki = 5620 nM T13201 CX3A0N 122192648 Ki = 3890 nM T13201 CU3F1V 122192649 Ki = 8910 nM T13201 CQ4NT8 122192650 Ki = 4270 nM T13201 C2REU8 122192651 Ki = 4310 nM T13201 CL5P4T 122192652 Ki = 5380 nM T13201 C0KF5I 122192653 Ki = 6520 nM T13201 CT64DB 122192654 Ki = 6530 nM T13201 CX05RY 122192671 Ki = 921 nM T13201 CE9ZC4 122192672 Ki > 10000 nM T13201 CUW2B9 122192673 Ki > 10000 nM T13201 CKU76Q 122192674 Ki = 210.7 nM T13201 C49KGU 122192675 Ki = 1568 nM T13201 CB0J2T 122192676 Ki = 239.5 nM T13201 CS63LF 122192677 Ki = 242.5 nM T13201 C4T3IO 122192678 Ki = 240.9 nM T13201 CTZ4L6 122192679 Ki = 172.8 nM T13201 C62VGD 122192680 Ki = 1243.2 nM T13201 CYND20 122192681 Ki = 2137.9 nM T13201 CLV5O9 122192682 Ki = 246.7 nM T13201 CH1N0C 122193189 Ki = 5230 nM T13201 C19HVL 122193190 Ki = 9620 nM T13201 C5TQJ1 122193251 Ki > 50000 nM T13201 C8XCL0 122193252 Ki = 3660 nM T13201 CH4IV8 122194771 Ki = 77 nM T13201 CQ7N0L 122194772 Ki = 78.8 nM T13201 CI5K2F 122194773 Ki = 67.5 nM T13201 CV51IU 122194774 Ki = 46.7 nM T13201 C7OFR6 122194775 Ki = 1635 nM T13201 C81HNW 122194776 Ki = 52.7 nM T13201 C8J5QV 122194777 Ki = 75.3 nM T13201 CV1C9T 122194778 Ki = 73.8 nM T13201 CJC1W3 122194779 Ki = 6.3 nM T13201 CU1TV5 122194780 Ki = 122 nM T13201 C4C1BE 122194781 Ki = 72.5 nM T13201 CR9I5Q 122194782 Ki = 236 nM T13201 C8SVY4 122194783 Ki = 80.1 nM T13201 C7HT8B 122194784 Ki = 8.9 nM T13201 CW8P3R 122194785 Ki = 70.5 nM T13201 COAK34 122194786 Ki = 589 nM T13201 CPN73S 122199224 Ki = 4860 nM T13201 CC1UO6 122226187 Ki = 15900 nM T13201 C7T0FH 122226188 Ki = 29100 nM T13201 C3EG2B 122226189 Ki = 49500 nM T13201 C18KAD 122367673 Ki = 3.75 nM T13201 CPN5F4 122367675 Ki = 0.54 nM T13201 C26IUP 122386532 Ki = 17100 nM T13201 CGE1Q6 122707121 Ki = 1178 nM T13201 C1JBF7 122707123 Ki = 35.2 nM T13201 CGPI62 123372490 Ki = 48.4 nM T13201 CV4GW7 126961712 Ki = 9.3 nM T13201 C0FD4E 126961713 Ki = 9.3 nM T13201 CD3HF0 127024855 Ki = 2.34 nM T13201 CXY79J 127024883 Ki > 10000 nM T13201 CK9C7T 127024884 Ki > 10000 nM T13201 C50MSQ 127024885 Ki > 10000 nM T13201 C4N6WJ 127024886 Ki = 2047 nM T13201 C5AES0 127024887 Ki > 10000 nM T13201 CHU95V 127024991 Ki > 10000 nM T13201 CP8O7D 127024992 Ki > 10000 nM T13201 CRHW31 127024993 Ki = 24.5 nM T13201 C57BLH 127025130 Ki = 68.4 nM T13201 C0T4VY 127025177 Ki = 5.45 nM T13201 CRTB63 127025292 Ki = 6965 nM T13201 CAO31Y 127025293 Ki = 6966 nM T13201 CL0ZR4 127025295 Ki > 10000 nM T13201 C9JNZ5 127025296 Ki = 83.6 nM T13201 C04USY 127025300 Ki = 137 nM T13201 CDB1Z9 127025301 Ki = 34.2 nM T13201 CYK6H1 127025302 Ki = 152 nM T13201 C7UF0B 127025480 Ki = 9717 nM T13201 CY7DI6 127025481 Ki = 1.7 nM T13201 C6M4SW 127025591 Ki > 10000 nM T13201 CUPA95 127025592 Ki = 3084 nM T13201 CWP36V 127025593 Ki = 12.5 nM T13201 C0DL8N 127026696 Ki = 3.6 nM T13201 C95QVS 127026977 Ki = 510 nM T13201 C09PAM 127026978 Ki = 871 nM T13201 CS96JF 127026979 Ki > 50000 nM T13201 CRB80M 127026980 Ki = 440 nM T13201 C0RBK5 127027010 Ki = 318 nM T13201 C0WY9H 127027097 Ki = 42.3 nM T13201 CP84DU 127027288 Ki = 370 nM T13201 CH30BV 127027289 Ki = 80.5 nM T13201 CM72RV 127027290 Ki = 66.9 nM T13201 CO3IJ7 127027291 Ki = 84 nM T13201 CTS74J 127027656 Ki = 3.09 nM T13201 CL9G1Y 127027664 Ki = 4.87 nM T13201 C9G5HM 127027733 Ki = 5.16 nM T13201 CT0E5I 127027734 Ki = 8.5 nM T13201 C2C3GA 127027735 Ki = 1.13 nM T13201 CT1Q7O 127027978 Ki = 3.63 nM T13201 CRL3B5 127028045 Ki = 2.77 nM T13201 C4O2XT 127028951 Ki > 10000 nM T13201 CFIW54 127029020 Ki = 656 nM T13201 C5RBS3 127029021 Ki = 2645 nM T13201 CPA6G5 127029022 Ki = 184.7 nM T13201 C74ZGJ 127029023 Ki = 370.3 nM T13201 CN3PH9 127029250 Ki > 10000 nM T13201 CTY1H9 127029498 Ki = 68.3 nM T13201 CC1E7F 127029514 Ki = 3.49 nM T13201 C1J0RU 127029568 Ki = 9 nM T13201 CE38AJ 127030670 Ki = 3.62 nM T13201 CKL6D3 127030963 Ki = 368 nM T13201 CWFJ07 127030973 Ki = 457 nM T13201 C4T2KL 127031264 Ki = 3.69 nM T13201 C8G3YC 127031289 Ki = 146 nM T13201 CHG8P6 127031292 Ki = 536 nM T13201 C8SA4R 127031846 Ki = 3.13 nM T13201 C2ILH1 127031859 Ki = 3.01 nM T13201 C4PZ0V 127032697 Ki = 259 nM T13201 CNH03L 127033707 Ki = 2.61 nM T13201 C8CN4T 127033708 Ki = 3.15 nM T13201 C1C8XD 127034555 Ki = 3.23 nM T13201 CC4J3A 127034556 Ki = 2.75 nM T13201 CO48QN 127034557 Ki = 2.84 nM T13201 CRN4X6 127034558 Ki = 3.01 nM T13201 CTAR42 127034559 Ki = 3.55 nM T13201 C67ZWL 127034560 Ki = 3.37 nM T13201 CS2K4U 127034999 Ki > 10000 nM T13201 CFG39M 127035855 Ki > 10000 nM T13201 C6MH2V 127035856 Ki > 10000 nM T13201 CVO4B6 127035857 Ki > 10000 nM T13201 CQC6P9 127035858 Ki > 10000 nM T13201 C7YA3N 127035859 Ki > 10000 nM T13201 CXZI89 127035860 Ki > 10000 nM T13201 C5KLP8 127035861 Ki > 10000 nM T13201 CTVN28 127036466 Ki = 68.9 nM T13201 CWPY69 127036947 Ki = 41.5 nM T13201 CL76JS 127037630 Ki > 10000 nM T13201 CY1JU3 127037755 Ki > 100 nM T13201 C0UQ7W 127037756 Ki > 10000 nM T13201 CQUE67 127037757 Ki = 4753 nM T13201 CL3Q0T 127037870 Ki > 10000 nM T13201 CK3VW1 127037881 Ki > 10000 nM T13201 CTSR32 127038212 Ki = 220 nM T13201 CQTS23 127038553 Ki = 9516 nM T13201 CG8B3V 127039153 Ki = 33.6 nM T13201 CIO74C 127039154 Ki = 41.3 nM T13201 C0L8NH 127039155 Ki = 46.8 nM T13201 CS96GU 127039479 Ki = 3540 nM T13201 C6WCG5 127039856 Ki = 285 nM T13201 C4NQ5H 127039905 Ki = 287 nM T13201 C3J8ET 127040041 Ki = 4368 nM T13201 C0P5HB 127040227 Ki = 81 nM T13201 CCD87Q 127040239 Ki = 315 nM T13201 C97DAS 127040240 Ki = 282 nM T13201 C9OZP8 127040553 Ki = 172 nM T13201 C4SH5D 127040554 Ki = 242 nM T13201 CCO9S8 127040555 Ki = 163 nM T13201 C12SMV 127041490 Ki = 1000 nM T13201 CSJ3V0 127041732 Ki = 7630 nM T13201 CG75VH 127041733 Ki = 6425 nM T13201 CQC6A4 127042329 Ki > 10000 nM T13201 CRZK01 127043469 Ki = 39.9 nM T13201 C41YOV 127044252 Ki = 33.9 nM T13201 CMTC13 127044428 Ki = 32.4 nM T13201 C7KU0Z 127044429 Ki = 35 nM T13201 CJO3U8 127044444 Ki = 87.6 nM T13201 CAXM67 127044445 Ki = 33.4 nM T13201 CHP23N 127044446 Ki > 40000 nM T13201 C1T4LU 127044499 Ki = 268 nM T13201 CI3PD8 127044664 Ki = 2954 nM T13201 CU5B2G 127044665 Ki = 1402 nM T13201 CM9QJ3 127044834 Ki = 150 nM T13201 C5HIY4 127044835 Ki = 28.5 nM T13201 CKW0B5 127044836 Ki = 42.3 nM T13201 C0KQB1 127044932 Ki = 3.2 nM T13201 C4WZJ7 127044997 Ki = 41.4 nM T13201 C1LIQ5 127044998 Ki = 104 nM T13201 C3S2GY 127044999 Ki = 34.3 nM T13201 C62OLS 127045037 Ki = 0.84 nM T13201 C31FCL 127045083 Ki = 702 nM T13201 CT9KP2 127045237 Ki = 6.5 nM T13201 C17GLC 127045238 Ki = 6.6 nM T13201 C1U0VA 127045339 Ki = 37.6 nM T13201 C5EX6R 127048632 Ki = 335.2 nM T13201 CG10PI 127048878 Ki = 862.42 nM T13201 C3PHY8 127048879 Ki = 299.73 nM T13201 COLX43 127048880 Ki = 295.77 nM T13201 CBJ74P 127048881 Ki = 3113.84 nM T13201 CK1X5H 127048994 Ki = 59.7 nM T13201 C2XK0I 127048995 Ki = 64.3 nM T13201 CY4P2X 127048996 Ki = 33.9 nM T13201 C6JB5S 127048997 Ki = 70.9 nM T13201 C1XE4W 127049197 Ki = 3227.77 nM T13201 CCX35L 127049198 Ki = 1896.08 nM T13201 CRE6O9 127049213 Ki = 272.62 nM T13201 CP40EB 127049242 Ki = 181 nM T13201 CLFB54 127049248 Ki = 225 nM T13201 C1T3WG 127049310 Ki = 47.7 nM T13201 CKO03S 127049970 Ki = 69 nM T13201 CP8KG9 127049971 Ki = 47.5 nM T13201 C5CNP8 127050174 Ki = 367.89 nM T13201 C9EJ6L 127050230 Ki = 88.7 nM T13201 CH07TV 127050456 Ki = 263.49 nM T13201 CP8U0D 127050457 Ki = 349.63 nM T13201 C65PAS 127050458 Ki = 1454.72 nM T13201 C7MI5Q 127050568 Ki = 48.8 nM T13201 C1RGQ6 127050569 Ki = 129.1 nM T13201 CB5W0L 127050570 Ki = 28.9 nM T13201 CUG58A 127050571 Ki = 94.5 nM T13201 CJP49X 127050777 Ki = 29.69 nM T13201 CER02F 127050778 Ki = 2001.23 nM T13201 CG17IO 127050812 Ki = 272 nM T13201 C8X6CY 127050822 Ki = 181 nM T13201 C9FZ4E 127050900 Ki = 40.3 nM T13201 C4IA5N 127051119 Ki = 221 nM T13201 CRDQ30 127051120 Ki = 180 nM T13201 CUWE95 127051804 Ki = 80.9 nM T13201 COBU26 127051805 Ki = 69 nM T13201 C7SIY6 127051806 Ki = 222.2 nM T13201 C5Y4DI 127051953 Ki = 192 nM T13201 CJ7WT3 127052106 Ki = 293.3 nM T13201 CM21NF 127052276 Ki = 21.95 nM T13201 C26TUM 127052712 Ki = 6.7 nM T13201 C7PS8D 127052713 Ki = 42.2 nM T13201 C32ART 127052714 Ki = 146.6 nM T13201 CI24ZM 127052900 Ki = 220.13 nM T13201 CEVZ36 127052901 Ki = 22.92 nM T13201 CX1Z2E 127052917 Ki = 310.48 nM T13201 CM8FI7 127052918 Ki = 315.19 nM T13201 CUOZ60 127052919 Ki = 272.94 nM T13201 C9D6CB 127053004 Ki = 42.4 nM T13201 CHN5K6 127567366 Ki = 84.5 nM T13201 C4JC3W 127573780 Ki = 513.6 nM T13201 C85FAK 129009671 Ki = 349.9 nM T13201 C7R6LY 129009672 Ki = 565.6 nM T13201 C2B6XM 129673327 Ki > 10000 nM T13201 CJC35Q 129856021 Ki > 10000 nM T13201 CCF61S 129883275 Ki = 208.6 nM T13201 CNB2M7 131839635 Ki = 6.7 nM T13201 C1V2RI 132353699 Ki = 85.9 nM T13201 C7Z4UB 132494202 Ki > 10000 nM T13201 CXN16P 132495328 Ki = 22 nM T13201 C20FGA 132495363 Ki > 500000 nM T13201 C4GR3Y 132498655 Ki = 37.9 nM T13201 CKLY32 132502995 Ki = 3745.9 nM T13201 CVM1A9 132547283 Ki = 243 nM T13201 C3H1NS 132547284 Ki = 849 nM T13201 C1FWS2 132547285 Ki = 276 nM T13201 C7Z5LX 132547286 Ki = 35.5 nM T13201 CW97YT 132547287 Ki = 318 nM T13201 CW18RT 132547288 Ki = 17.9 nM T13201 COC54I 132547289 Ki = 97.5 nM T13201 CX4DM9 132547290 Ki = 79.8 nM T13201 C5JM7W 132547291 Ki = 83.3 nM T13201 C7V6XS 132547292 Ki = 64.3 nM T13201 C5O1JE 132547793 Ki > 100000 nM T13201 CKYC42 132547798 Ki = 80100 nM T13201 C7MZ8T 132569639 Ki = 3790 nM T13201 CRL24F 132596304 Ki = 8914 nM T13201 C6OA8Z 132819872 Ki = 983 nM T13201 CJGH58 132819873 Ki = 716 nM T13201 COT92G 132819874 Ki = 4250 nM T13201 COS36W 132819875 Ki = 826 nM T13201 CMAU69 132819876 Ki = 737 nM T13201 CY62CQ 132938107 Ki = 387 nM T13201 CB8T7K 132938108 Ki = 169 nM T13201 CY6L7Z 132941396 Ki = 876 nM T13201 C4K1YW 132961363 Ki = 13.6 nM T13201 CQ64ZM 132961364 Ki = 3661 nM T13201 C5LGV6 132961365 Ki = 96.1 nM T13201 CD9ET2 132961426 Ki = 49.2 nM T13201 CR80OW 132961427 Ki = 179 nM T13201 C17QYW 132961557 Ki = 8.7 nM T13201 CGC58D 132961558 Ki = 5.4 nM T13201 CZDR23 132961559 Ki = 96 nM T13201 C4Y5SW 132961560 Ki = 52.9 nM T13201 CXF7N2 132961561 Ki = 4.9 nM T13201 CQAC41 132961562 Ki = 25.3 nM T13201 C57MKX 132961563 Ki = 40 nM T13201 C6N1PW 132961564 Ki = 90.7 nM T13201 CZ60IC 132961565 Ki = 8.8 nM T13201 CEP32W 132991412 Ki > 10000 nM T13201 C69NDK 133107891 Ki = 5.2 nM T13201 C2AIR8 134129901 Ki = 67.4 nM T13201 C1Y9AL 134130029 Ki = 23.9 nM T13201 CG0HL2 134130044 Ki = 218 nM T13201 C63CQL 134130121 Ki = 943 nM T13201 CU10DE 134130177 Ki = 84.5 nM T13201 C82HUT 134130285 Ki = 624 nM T13201 CMZ76O 134130322 Ki = 9695 nM T13201 CP8XK0 134130364 Ki = 49.7 nM T13201 C8AL2D 134130377 Ki = 500 nM T13201 C7N0JD 134130389 Ki = 662 nM T13201 C83LZE 134130471 Ki = 390 nM T13201 C5N8AO 134130483 Ki = 293.8 nM T13201 C9V3LX 134130512 Ki = 45.8 nM T13201 CO7G6J 134130566 Ki = 8.2 nM T13201 C69IZA 134130639 Ki > 10000 nM T13201 C8MGN3 134130817 Ki = 6376.6 nM T13201 C52IRH 134131086 Ki = 40.9 nM T13201 CZ7CA3 134131127 Ki = 510 nM T13201 C9HVL2 134131189 Ki = 7.5 nM T13201 C5XU9Y 134131319 Ki = 9330 nM T13201 C7GBW5 134131361 Ki = 60.5 nM T13201 CZ2YK7 134131524 Ki = 9510 nM T13201 C3WJR8 134131535 Ki = 41.8 nM T13201 CQ0K5P 134131567 Ki = 7.3 nM T13201 C8Q5JZ 134131574 Ki = 917 nM T13201 CUVB06 134131580 Ki = 287 nM T13201 C94HZF 134131659 Ki = 7.9 nM T13201 CU5B8H 134131865 Ki = 351.1 nM T13201 CZQ3T2 134132041 Ki > 10000 nM T13201 C89TVU 134132755 Ki = 4762.2 nM T13201 C2UIM6 134132835 Ki = 683 nM T13201 CECZ43 134133137 Ki > 500000 nM T13201 CFQG76 134133776 Ki = 286.8 nM T13201 CT8Z2Q 134133785 Ki = 774.7 nM T13201 C83QKJ 134133977 Ki = 92.8 nM T13201 CM3J9G 134134653 Ki = 295 nM T13201 CJ3EQ2 134136523 Ki = 949.8 nM T13201 CHR23F 134137004 Ki > 10000 nM T13201 C4IO1K 134137058 Ki = 2470 nM T13201 C2X1UG 134137145 Ki = 50.1 nM T13201 CHM19B 134139215 Ki = 2860.6 nM T13201 CWG0L5 134139228 Ki = 278.1 nM T13201 CRNF42 134140829 Ki = 6529.5 nM T13201 C1T9JU 134140936 Ki = 475.8 nM T13201 CG4NU1 134141378 Ki = 402 nM T13201 CJ4R6E 134141819 Ki > 500000 nM T13201 CDUW03 134142004 Ki = 706 nM T13201 CC05JV 134142010 Ki = 683 nM T13201 CIK25S 134142323 Ki = 2419.8 nM T13201 CIRG86 134142877 Ki = 5910.6 nM T13201 CWT6O9 134142989 Ki = 7469.6 nM T13201 C5BD1C 134143174 Ki > 10000 nM T13201 CWQ62J 134144541 Ki > 10000 nM T13201 CG7X9K 134144756 Ki = 495.2 nM T13201 CJ5QD3 134144926 Ki = 7295.2 nM T13201 CR5F8T 134145685 Ki = 2868.4 nM T13201 CBK73M 134146037 Ki = 512.6 nM T13201 C8FV5Y 134147016 Ki > 10000 nM T13201 C0TV9S 134147261 Ki = 661.7 nM T13201 CDH38B 134147400 Ki > 10000 nM T13201 CDSM29 134147656 Ki = 1870 nM T13201 C85ABV 134147911 Ki = 3941.1 nM T13201 CGBZ05 134148709 Ki = 63.8 nM T13201 CS7K8C 134149271 Ki = 3654.6 nM T13201 C1Q8GK 134149666 Ki = 195.7 nM T13201 CF31OS 134149711 Ki = 1280 nM T13201 CD5TI1 134149815 Ki = 9260.9 nM T13201 CZ2C3J 134149835 Ki = 59.8 nM T13201 C2NXB7 134151324 Ki = 3600 nM T13201 CIL4H9 134151823 Ki > 10000 nM T13201 C9GF7L 134152087 Ki = 473.3 nM T13201 CR4VE0 134152281 Ki > 500000 nM T13201 CU0T4X 134152542 Ki = 406.8 nM T13201 CZ9C1N 134152694 Ki = 965 nM T13201 CZ4WI8 134152920 Ki = 8704.7 nM T13201 C4WBC6 134153047 Ki = 123 nM T13201 CD4EN0 134153199 Ki = 3688 nM T13201 CH6OT4 134153506 Ki = 404.8 nM T13201 CZ9T6I 134153525 Ki > 10000 nM T13201 CWSI54 134154346 Ki = 1579.4 nM T13201 CSK6L9 134154625 Ki > 500000 nM T13201 CQZU97 134154945 Ki > 10000 nM T13201 CCU96S 134155195 Ki = 910 nM T13201 CG69UV 134155483 Ki > 500000 nM T13201 C52UTP 134156470 Ki = 359.7 nM T13201 C7OV6T 134156655 Ki = 2962.3 nM T13201 CZ9L5F 134158397 Ki = 8.8 nM T13201 CR3Q5U 134159783 Ki = 293.5 nM T13201 CV9W6N 134159784 Ki = 21.9 nM T13201 C8C0TO 134812637 Ki = 811.8 nM T13201 CV9X5Y 134817795 Ki = 49.4 nM T13201 C19BHQ 134817796 Ki = 273.3 nM T13201 CY3E4D 134817797 Ki = 306.1 nM T13201 C8IF6V 134817798 Ki = 255.1 nM T13201 C0UL7A 134828600 Ki = 5200 nM T13201 C4ZLP6 134828601 Ki = 690 nM T13201 C3OLP6 134828602 Ki = 7580 nM T13201 CJT9W0 135393499 Ki = 1.7 nM T13201 CK8FP3 135393500 Ki = 9.3 nM T13201 CRL4V7 135393501 Ki = 0.69 nM T13201 C19SUQ 135405876 Ki > 10000 nM T13201 CTR37Z 135408753 Ki > 500000 nM T13201 C6QT0M 135411191 Ki = 1000 nM T13201 C4TCL7 135411929 Ki = 422 nM T13201 C3YE2K 135412032 Ki > 10000 nM T13201 CW9B7C 135422576 Ki = 91.9 nM T13201 C4CXD1 135434964 Ki = 467.3 nM T13201 CFK9A4 135434965 Ki = 1810.2 nM T13201 CY7RT4 135442220 Ki = 8020 nM T13201 CKAF26 135460193 Ki = 32 nM T13201 C1KUG5 135495066 Ki = 355000 nM T13201 C7E6AM 135496540 Ki = 378 nM T13201 C3MV2E 135519301 Ki = 10500 nM T13201 CPW4T3 135530880 Ki = 81.5 nM T13201 C0WEU9 135537166 Ki = 229 nM T13201 C7E8RX 135570228 IC50 = 2.13 nM T13201 CC8IO3 135595465 Ki = 454 nM T13201 C74TBX 135595467 Ki = 384 nM T13201 C8D6XA 135595468 Ki = 70 nM T13201 CX1NF7 135595474 Ki = 351 nM T13201 CL71ND 135645043 Ki > 50000 nM T13201 CHM06N 135794287 Ki = 5950 nM T13201 C6J2RU 135878387 IC50 = 374 nM T13201 C1WH3Z 135891810 Ki = 59 nM T13201 CSH8M1 135995959 Ki = 41 nM T13201 CB90PQ 135995960 Ki = 7.5 nM T13201 C47ART 136002512 IC50 = 80 nM T13201 C2J5FZ 136002546 IC50 = 120 nM T13201 CJ31YP 136002685 IC50 = 140 nM T13201 C0T8LG 136002686 IC50 = 100 nM T13201 CXD6J2 136002687 IC50 = 550 nM T13201 CNG0L4 136044222 Ki = 4320 nM T13201 CQ02AW 136044223 Ki = 5335 nM T13201 C47KQP 136053622 Ki = 463 nM T13201 C1M7DN 136053656 Ki = 387 nM T13201 C8CV0N 136056550 Ki = 105 nM T13201 CFT0H2 136059729 IC50 = 80 nM T13201 C31CEK 136094773 Ki = 0.85 nM T13201 C3VG8C 136094774 Ki = 7.6 nM T13201 C38LKD 136104491 Ki = 51630 nM T13201 C0PNH7 136104492 Ki = 3710 nM T13201 CNW21F 136104493 Ki = 8030 nM T13201 CST63W 136104494 Ki = 3340 nM T13201 C9GQS8 136104495 Ki = 7890 nM T13201 CHG82O 136118030 Ki = 620 nM T13201 C4KH2F 136138702 Ki = 5.1 nM T13201 C4A2XS 136198631 Ki = 398.78 nM T13201 C93PWB 136198632 Ki > 10000 nM T13201 CVME35 136198643 Ki = 448 nM T13201 CZ9M6L 136217534 Ki = 318 nM T13201 C8Q9ES 136217535 Ki = 448 nM T13201 CIX3N6 136217536 Ki = 1079 nM T13201 CBO5I1 136242872 Ki = 83 nM T13201 CQDT25 136242873 Ki = 48 nM T13201 CK5AZ7 136242878 Ki = 34 nM T13201 C1NTA3 136418497 Ki = 8484.3 nM T13201 CQUV48 136499038 Ki = 92 nM T13201 C6VS7N 136607460 Ki = 80.4 nM T13201 CAC75Q 136607461 Ki = 126 nM T13201 CYKW91 136728963 Ki = 92.5 nM T13201 CI28TM 136934908 Ki = 421 nM T13201 C9UKC8 136998786 Ki = 4400 nM T13201 C3QFS1 136998787 Ki = 4235 nM T13201 C1P9FJ 136998788 Ki = 1750 nM T13201 CZ40LF 137028501 Ki = 53.7 nM T13201 C5Q8PD 137028502 Ki = 102 nM T13201 CSL47A 137028503 Ki = 9 nM T13201 C7T1HR 137028504 Ki = 52.4 nM T13201 C9WH2P 137028505 Ki = 9.7 nM T13201 CGBQ10 137028506 Ki = 38.3 nM T13201 C4DHG6 137028507 Ki = 6.7 nM T13201 CIP84X 137028508 Ki = 7.6 nM T13201 CF14KA 137028511 Ki = 49.5 nM T13201 CXHB30 137028512 Ki = 61.9 nM T13201 CRMC05 137028513 Ki = 5.7 nM T13201 CJH4E5 137028514 Ki = 7.1 nM T13201 CGAR93 137028515 Ki = 5.2 nM T13201 C4QG2K 137028516 Ki = 7.1 nM T13201 C2GMH5 137028517 Ki = 70.4 nM T13201 CBX6S7 137028518 Ki = 14.9 nM T13201 C52OFD 137028519 Ki = 510 nM T13201 CUW85H 137062187 Ki = 85.9 nM T13201 C4XY9S 137091066 Ki = 679 nM T13201 C64ITR 137091070 Ki = 894 nM T13201 C0BEH8 137093138 Ki = 428 nM T13201 CD6C0A 137093141 Ki = 567 nM T13201 CJI35T 137124112 Ki = 652 nM T13201 CJI47D 137175023 Ki = 295 nM T13201 CM70RT 137175046 Ki = 579 nM T13201 CVZR36 137175050 Ki = 375 nM T13201 CCG5D7 137175057 Ki = 816 nM T13201 COFC53 137175058 Ki = 600 nM T13201 CV57WL 137175059 Ki = 778 nM T13201 CM1FL4 137175099 Ki = 249 nM T13201 CR6U9I 137175102 Ki = 490 nM T13201 CHK1L6 137175124 Ki = 742 nM T13201 CK2M1V 137175125 Ki = 426 nM T13201 CCP87O 137175126 Ki = 539 nM T13201 C4WZ5F 137175214 Ki = 414 nM T13201 CJ2DW1 137196867 Ki = 554.4 nM T13201 CUJ3N2 137196890 Ki = 76.1 nM T13201 CE9QV3 137226330 Ki = 22.5 nM T13201 C4SMA5 137226331 Ki = 37.1 nM T13201 C2H6VC 137226372 Ki = 462 nM T13201 CZY9D7 137226374 Ki = 95.6 nM T13201 C6YBD3 137226375 Ki = 9 nM T13201 C7DMR8 137226384 Ki = 62.8 nM T13201 C2KG3D 137226385 Ki = 45.2 nM T13201 C0KMB4 137226399 Ki = 9.2 nM T13201 CD1VC9 137226400 Ki = 7.9 nM T13201 C4F8NU 137226401 Ki = 10.2 nM T13201 CW65FQ 137226402 Ki = 8.5 nM T13201 CY95JF 137226420 Ki = 29.3 nM T13201 CM58FB 137228156 Ki = 6.4 nM T13201 CK94PV 137228157 Ki = 41 nM T13201 CAY48F 137228158 Ki = 7.9 nM T13201 COW81G 137273278 Ki = 901 nM T13201 CY3P7J 137283379 Ki = 19.1 nM T13201 CPM09K 137287437 Ki = 13.05 nM T13201 CNS38T 137287438 Ki = 9.88 nM T13201 C1G8YE 137287439 Ki = 14.47 nM T13201 C1BOM7 137287440 Ki = 13.25 nM T13201 CY4K2R 137287441 Ki = 24.4 nM T13201 C39QNK 137287442 Ki = 21.88 nM T13201 CW52IQ 137631447 Ki = 2.29 nM T13201 CRK6Y9 137631731 Ki = 3221 nM T13201 CZ5GQ4 137631746 Ki > 100 nM T13201 CFQ5W2 137631798 Ki > 50000 nM T13201 CRHD41 137632004 IC50 = 0.699 nM T13201 C7O3CP 137632017 Ki = 3.11 nM T13201 C83VZC 137632115 Ki = 3020 nM T13201 CBJ75C 137632178 Ki = 745.6 nM T13201 CN8UL1 137632214 Ki = 0.99 nM T13201 CYD0E3 137632442 Ki = 85.7 nM T13201 CL5K3D 137632743 Ki > 100 nM T13201 CE20FG 137632898 Ki = 4.76 nM T13201 CO25DP 137632949 Ki = 275.6 nM T13201 C9YKD5 137633039 Ki = 523.7 nM T13201 CFE79H 137633320 Ki > 10000 nM T13201 C5J3AX 137633409 Ki = 316 nM T13201 C9AD2H 137633797 Ki = 2330 nM T13201 CVNO32 137633860 Ki = 221.8 nM T13201 C4CIT3 137634087 Ki = 6820 nM T13201 C5NLG4 137634142 Ki = 8710 nM T13201 C7N0ER 137634525 Ki = 75900 nM T13201 C0P6ZT 137634762 Ki = 924.9 nM T13201 CZHO28 137634971 IC50 = 0.518 nM T13201 CP0EC3 137635051 Ki = 615.8 nM T13201 C08ANJ 137635055 Ki = 5520 nM T13201 CY1HI4 137635059 Ki = 775 nM T13201 C4YV1N 137635125 Ki = 698 nM T13201 C3NQ9Y 137635300 Ki = 95.7 nM T13201 C1ZKU2 137635320 Ki = 81.6 nM T13201 CS6M2N 137635469 Ki > 10000 nM T13201 CDB92Z 137635478 IC50 = 0.535 nM T13201 CNJV53 137635486 Ki = 5.83 nM T13201 CVNX12 137635652 Ki = 650 nM T13201 CZ4Q1T 137636083 Ki = 3200 nM T13201 C9GIX7 137636130 Ki = 1.48 nM T13201 CV12YX 137636350 Ki > 100 nM T13201 CE46DY 137636432 Ki = 563 nM T13201 CK0N2Y 137636453 Ki = 264 nM T13201 C5R7LW 137636489 IC50 = 0.57 nM T13201 CM9YC2 137636494 Ki > 10000 nM T13201 CLR6U5 137636505 Ki = 435 nM T13201 C3PXL8 137636591 IC50 = 1.69 nM T13201 C5D3BS 137636775 Ki = 7420 nM T13201 CMX9T3 137636945 Ki = 0.81 nM T13201 C7YKB0 137636981 Ki = 3300 nM T13201 C2Z7GO 137637071 Ki = 38.9 nM T13201 C0H2CK 137637173 Ki = 66.3 nM T13201 CWO5Z6 137637365 Ki > 100 nM T13201 CGV9M8 137637508 Ki > 10000 nM T13201 CG0N8K 137637564 Ki = 384.5 nM T13201 CQ5K1H 137637688 Ki = 4600 nM T13201 C80KCO 137637736 Ki = 3603.7 nM T13201 C2HY8G 137637767 Ki = 245 nM T13201 CB3KA0 137638304 Ki = 624.2 nM T13201 CHQ3P9 137638456 Ki = 42 nM T13201 CK6OW4 137638637 Ki = 15.6 nM T13201 C6V8ED 137638882 Ki = 16 nM T13201 C64JQN 137639095 Ki = 6.9 nM T13201 CVJ35I 137639180 Ki = 5.97 nM T13201 C12QYH 137639189 Ki = 8.59 nM T13201 C4LB2X 137639339 Ki = 61.5 nM T13201 CX7TE5 137639357 Ki = 744 nM T13201 C0IQ1U 137639377 Ki = 3347 nM T13201 C29XAH 137639434 Ki = 8390.6 nM T13201 C8DW0G 137639460 IC50 = 0.677 nM T13201 CV4L6A 137639464 IC50 = 0.56 nM T13201 CH2C3F 137639611 Ki = 619.6 nM T13201 CPR04H 137639655 Ki = 3570 nM T13201 C4SP7Q 137639785 Ki = 83.9 nM T13201 COE61G 137639833 Ki = 81300 nM T13201 C2OT9R 137640310 Ki = 3490 nM T13201 C5OU2V 137640459 Ki = 3095.2 nM T13201 CX3JI9 137640517 Ki = 73.3 nM T13201 CZGW35 137640627 Ki = 9160 nM T13201 CQN3L7 137640789 Ki = 0.12 nM T13201 C8P3SC 137640892 Ki > 10000 nM T13201 CJ4M2A 137640917 Ki = 781.4 nM T13201 CR65OQ 137640944 Ki = 64.7 nM T13201 C75WMG 137641075 Ki = 6140 nM T13201 C6B0CQ 137641198 Ki = 2.2 nM T13201 C0HER8 137641290 Ki = 909 nM T13201 CR2MU6 137641422 Ki = 2.91 nM T13201 CMOZ57 137641425 Ki = 5900 nM T13201 C4FN0Q 137641666 Ki = 882 nM T13201 C53ZAF 137641717 Ki > 10000 nM T13201 CR5JZ8 137642047 Ki > 10000 nM T13201 CCSN50 137642054 Ki > 100 nM T13201 CN6WS9 137642180 Ki = 1771 nM T13201 C0Z9DH 137642233 Ki = 2.18 nM T13201 C6YV7B 137642310 Ki = 850 nM T13201 CEOC90 137642331 Ki = 7255 nM T13201 CSY67B 137642513 Ki = 675.5 nM T13201 C51DEC 137642551 IC50 = 0.556 nM T13201 C61TSP 137642864 Ki > 100000 nM T13201 C7ZX8Q 137643203 Ki = 4.17 nM T13201 C3Y2GU 137643607 Ki = 92.3 nM T13201 C1BW5I 137643671 Ki = 89800 nM T13201 CZ1W3N 137643790 IC50 = 0.903 nM T13201 C0B8QA 137643949 Ki > 100 nM T13201 CG13TO 137643998 Ki = 6.28 nM T13201 CF31BQ 137644307 Ki = 93.9 nM T13201 CI4A9L 137644641 Ki = 9350 nM T13201 CIK49D 137644678 Ki = 47.8 nM T13201 CV75NJ 137644865 Ki > 10000 nM T13201 CFA3R0 137644914 Ki = 4450.2 nM T13201 CWQ91B 137644949 Ki = 276 nM T13201 CHG72J 137644957 Ki = 425 nM T13201 CV0AH9 137645517 Ki = 293 nM T13201 C6UAB5 137645654 Ki = 844.5 nM T13201 CDZ6T8 137645734 Ki = 875.4 nM T13201 CFV6T3 137645790 Ki = 3.36 nM T13201 C3CI0M 137645793 Ki = 768.6 nM T13201 CBRK83 137645944 Ki = 73.8 nM T13201 C7E6NL 137646223 Ki = 1730 nM T13201 C4WOE0 137646284 Ki = 441 nM T13201 C10YVU 137646329 Ki = 1790 nM T13201 C5WG2P 137646543 Ki = 149.4 nM T13201 CO3V9P 137646707 IC50 = 0.29 nM T13201 C0YFX2 137646956 Ki > 10000 nM T13201 CVE3K2 137647149 IC50 = 0.346 nM T13201 CRP78K 137647221 Ki > 100 nM T13201 C5T2VN 137647270 Ki = 7370 nM T13201 CXD9A0 137647636 Ki = 3.5 nM T13201 CR2H7M 137647845 Ki = 860 nM T13201 CY15KD 137648125 Ki = 262 nM T13201 C5PEA6 137648128 Ki = 7650 nM T13201 CA56EB 137648145 IC50 = 0.624 nM T13201 CCD71U 137648259 Ki = 9381.1 nM T13201 C49PLO 137648279 Ki = 6149.3 nM T13201 CW8CL7 137648379 Ki = 44.7 nM T13201 CU81DA 137648494 Ki = 719 nM T13201 CK14XO 137648525 Ki = 4152 nM T13201 C21TVD 137648644 Ki = 872.9 nM T13201 C6RIM2 137648717 Ki = 845.2 nM T13201 C6IB1L 137648807 Ki = 558 nM T13201 C82NJP 137648964 Ki = 8.51 nM T13201 CEZT03 137649001 Ki = 802.5 nM T13201 CI9LS2 137649321 Ki = 64.1 nM T13201 CY94BR 137649373 Ki = 9040 nM T13201 CSWR71 137649376 Ki = 781.3 nM T13201 C7PEQ0 137649468 IC50 = 4.21 nM T13201 CY0QB6 137649527 IC50 = 0.45 nM T13201 CGLM50 137649870 Ki = 164 nM T13201 C2HA7Q 137649882 Ki > 10000 nM T13201 C4N1MP 137650156 Ki = 850 nM T13201 CCZ4N1 137650188 Ki = 91.3 nM T13201 C1FO3T 137650198 Ki = 296 nM T13201 C91KQA 137650256 Ki = 143 nM T13201 CD08YK 137650293 Ki = 514.9 nM T13201 CKJ36G 137650647 Ki = 521.2 nM T13201 CD7S5L 137650698 Ki > 100000 nM T13201 CJV8Q6 137650823 Ki = 201 nM T13201 CV89IF 137651491 Ki = 255.9 nM T13201 C5V6XP 137651635 Ki = 135 nM T13201 CSTP12 137651755 Ki = 5.6 nM T13201 C01BXO 137651769 Ki > 100 nM T13201 CY0C6Z 137652226 Ki > 100 nM T13201 C6GWB1 137652305 Ki > 100 nM T13201 CN3RQ8 137652373 Ki > 10000 nM T13201 C5DG1K 137652445 Ki = 4435 nM T13201 CP4GY0 137652940 Ki = 2640 nM T13201 C03TAW 137653117 Ki = 6640 nM T13201 CN0W6U 137653170 Ki > 50000 nM T13201 C9UGN4 137653309 Ki = 8130 nM T13201 C45WNI 137653361 Ki = 4.49 nM T13201 C8Y7XR 137653485 Ki = 9.6 nM T13201 CIV3E9 137653528 Ki = 85.7 nM T13201 C4U9KA 137653686 Ki = 2.91 nM T13201 C0O3JI 137654169 Ki = 1190 nM T13201 CTP0U2 137654343 Ki = 667.9 nM T13201 CNJ6P9 137654601 Ki > 10000 nM T13201 CS3LD8 137654917 Ki = 2650 nM T13201 CRC23M 137655132 Ki = 73 nM T13201 CWT49Q 137655252 Ki = 5670 nM T13201 CXC7I2 137655261 Ki = 206.2 nM T13201 C2P5FH 137655445 Ki = 680 nM T13201 C3DT7S 137655450 Ki > 100 nM T13201 CASB61 137655528 Ki > 100 nM T13201 C0XPN2 137655580 Ki = 177.8 nM T13201 CUO84H 137655694 Ki > 10000 nM T13201 CAZ27T 137655913 Ki = 89.9 nM T13201 C27ALW 137655946 Ki = 65.6 nM T13201 CC0OY9 137655984 Ki = 64.9 nM T13201 C8TJN9 137656061 Ki = 3649 nM T13201 CHD58S 137656247 Ki > 10000 nM T13201 COEY05 137656447 Ki = 264.9 nM T13201 CRXD65 137656549 Ki = 3.16 nM T13201 C06ONV 137656670 Ki = 57.6 nM T13201 C0CK7G 137656796 Ki = 8550.9 nM T13201 CG5EK0 137656938 Ki > 10000 nM T13201 CT7CW2 137657041 Ki = 6.15 nM T13201 C3PAQ7 137657121 Ki > 10000 nM T13201 C2SYC9 137657578 Ki = 543 nM T13201 C8RNZ6 137657759 Ki > 100 nM T13201 C0KI6G 137657917 Ki = 673.7 nM T13201 CTI2V7 137658103 Ki > 10000 nM T13201 CT5PO9 137658239 Ki = 7290 nM T13201 CH39CL 137658251 Ki = 348 nM T13201 C3W4BA 137658271 Ki = 484 nM T13201 C41MLN 137658275 Ki > 10000 nM T13201 CKX78V 137658314 Ki = 8702 nM T13201 CL2H0T 137658375 Ki > 100 nM T13201 CMR2L9 137658572 IC50 = 0.77 nM T13201 C7V6MY 137658589 Ki = 1650 nM T13201 CT98MV 137658877 Ki > 100 nM T13201 C8YV5D 137659052 Ki = 3.4 nM T13201 CXO9Y7 137659205 Ki > 100 nM T13201 CE3VX9 137659225 IC50 = 0.29 nM T13201 CJ5O8M 137659269 Ki = 3390 nM T13201 CO1RD4 137659342 Ki = 5500 nM T13201 C5AM2K 137659383 Ki > 10000 nM T13201 C40MRZ 137659514 Ki = 3.73 nM T13201 CCX48V 137659570 Ki = 436 nM T13201 C4MB7C 137659778 Ki = 481 nM T13201 CXK83H 137659797 Ki = 4975.9 nM T13201 CHKB25 137659801 Ki > 10000 nM T13201 CSPB10 137659919 Ki = 68.8 nM T13201 C60DEN 137660288 Ki > 10000 nM T13201 CMS92X 137660799 Ki = 734.2 nM T13201 C0TZD5 137661006 Ki > 100000 nM T13201 C0PIE6 137661027 Ki = 792.3 nM T13201 CQ56MJ 137661167 Ki = 899.4 nM T13201 C62QWK 137661307 Ki = 5817 nM T13201 CF6Z9A 137661353 Ki = 965 nM T13201 CRC92Y 137661359 Ki = 10.9 nM T13201 CN1JH4 137661469 Ki = 383.7 nM T13201 C1Z8KG 137661675 Ki = 9.3 nM T13201 C03HGD 137661687 Ki = 0.12 nM T13201 COA7Q3 137661801 IC50 = 0.28 nM T13201 C74YSR 137661914 Ki = 90.5 nM T13201 CEAR56 137662187 Ki = 3060 nM T13201 CMP8S7 137662201 Ki = 7488 nM T13201 CFR73V 137662256 Ki > 10000 nM T13201 CO8UE3 137662293 Ki = 2988.1 nM T13201 CTK0L9 137662315 IC50 = 0.288 nM T13201 C08ZTR 138393077 Ki = 441 nM T13201 CIX41M 138393379 Ki = 140.6 nM T13201 C7V9ZF 138455154 Ki = 7.3 nM T13201 CBOM51 138753317 Ki = 237.2 nM T13201 CB83JY 139593608 Ki = 48.7 nM T13201 C8TWF0 139597735 Ki = 4350 nM T13201 CR10ZH 139823666 Ki > 1000 nM T13201 C78UAW 142468585 Ki = 81.6 nM T13201 CZY8Q6 142468589 Ki = 2.2 nM T13201 C3HMI0 142468591 Ki = 1570 nM T13201 CHA65U 142468595 Ki > 50000 nM T13201 C6KE9A 142468600 Ki > 50000 nM T13201 C65DHJ 142468602 Ki = 9.1 nM T13201 CI02LX 142468604 Ki = 3930 nM T13201 C7LP3J 142468605 Ki > 50000 nM T13201 CA9O2I 142468608 Ki = 619 nM T13201 CUE58A 142547533 Ki > 10000 nM T13201 C6GB9T 143032987 Ki > 10000 nM T13201 CNW7H1 145948231 Ki = 63 nM T13201 C3PF4Q 145948234 Ki = 52.5 nM T13201 C7Y8GF 145949148 Ki = 570 nM T13201 CQC2D5 145949182 Ki = 60.7 nM T13201 C0Z2WP 145949184 Ki = 6.6 nM T13201 CI9H2E 145949226 Ki > 10000 nM T13201 CK65AC 145949290 Ki = 4721.4 nM T13201 C8BZI0 145949366 Ki = 316 nM T13201 CP6AM5 145949377 Ki = 8.9 nM T13201 CHVR98 145949393 Ki = 8084.3 nM T13201 CGLD54 145949403 Ki > 10000 nM T13201 C3LZH7 145949437 Ki = 645.5 nM T13201 CROP78 145949554 Ki = 59.1 nM T13201 C09ZGW 145949615 Ki > 10000 nM T13201 CA01QK 145949650 Ki = 37.7 nM T13201 C7I3GC 145949670 Ki = 894.2 nM T13201 C7X0DZ 145949728 Ki = 2578 nM T13201 CIU2Y1 145949743 Ki = 66.5 nM T13201 CA05JL 145949806 Ki = 34.2 nM T13201 CHI5L3 145949836 Ki = 29.5 nM T13201 C3U1AB 145949909 Ki = 37.2 nM T13201 C20RXT 145949974 Ki = 193.8 nM T13201 CJ8R3M 145950033 Ki = 455.7 nM T13201 CSW7B8 145950055 Ki > 10000 nM T13201 CISR74 145950124 Ki = 82.8 nM T13201 CRH3U4 145950259 Ki = 288 nM T13201 C7DBT4 145950298 Ki > 10000 nM T13201 CO9UN4 145950340 Ki = 42.6 nM T13201 CW56LV 145950373 Ki = 63.9 nM T13201 CJSK40 145950390 Ki > 10000 nM T13201 C2H9QY 145950512 Ki = 513.8 nM T13201 C7BK9O 145950527 Ki = 385.6 nM T13201 C63SMQ 145950568 Ki > 10000 nM T13201 CE58JF 145950709 Ki = 7148.1 nM T13201 C0C9FT 145950755 Ki = 426.2 nM T13201 C8XAH1 145950880 Ki = 6.9 nM T13201 C53EGH 145950894 Ki = 6.6 nM T13201 CRD27H 145950965 Ki = 29 nM T13201 C8IGY9 145950981 Ki > 10000 nM T13201 C9QUL0 145951028 Ki = 93 nM T13201 C1X2FW 145951066 Ki = 548 nM T13201 C7W5PI 145951214 Ki = 83.6 nM T13201 C87JIM 145951255 Ki = 350.4 nM T13201 CJ6LR3 145951259 Ki = 318 nM T13201 CPD05I 145951366 Ki = 297.1 nM T13201 C7LMU1 145951380 Ki = 30.7 nM T13201 C86DBE 145951463 Ki = 466.1 nM T13201 CB8V7M 145951488 Ki = 54.4 nM T13201 CL25SI 145951508 Ki > 10000 nM T13201 CS8GO6 145951628 Ki = 355 nM T13201 C38QHU 145951654 Ki = 70.7 nM T13201 CIM8X0 145951670 Ki = 127.2 nM T13201 CH9J8K 145951685 Ki = 22.1 nM T13201 C74RDJ 145951698 Ki = 64.5 nM T13201 CJ2W6V 145951720 Ki = 7.3 nM T13201 CZ23SB 145951758 Ki = 3133.7 nM T13201 CC0P1U 145951787 Ki > 10000 nM T13201 CN4MW7 145951794 Ki = 450 nM T13201 CF20QP 145951819 Ki = 51.6 nM T13201 C98SYV 145951855 Ki = 4871 nM T13201 CQC79A 145951865 Ki = 230.6 nM T13201 C2OTU3 145951886 Ki = 755.4 nM T13201 CF7U3J 145951902 Ki = 574 nM T13201 CKZT53 145951931 Ki > 10000 nM T13201 C3R8NQ 145951979 Ki = 3341 nM T13201 CGFU20 145952201 Ki > 10000 nM T13201 C4N3QL 145952239 Ki = 148.6 nM T13201 CUJ2G6 145952345 Ki = 20.2 nM T13201 CM30EN 145952365 Ki = 841.1 nM T13201 CU69PG 145952370 Ki = 395.9 nM T13201 C75RDX 145952490 Ki = 352.2 nM T13201 CP92AH 145952604 Ki = 1924.4 nM T13201 C26OLK 145952634 Ki = 5995 nM T13201 CW42HX 145952649 Ki = 70.2 nM T13201 C49OWE 145952696 Ki = 639 nM T13201 CWE6M8 145952775 Ki > 10000 nM T13201 C81UYG 145952794 Ki = 8.7 nM T13201 C6PZ3H 145952834 Ki = 67.7 nM T13201 CK4Q0X 145952846 Ki = 295.7 nM T13201 C56QVF 145952880 Ki = 228.8 nM T13201 CAS8M7 145952940 Ki = 274.5 nM T13201 CUB49H 145952983 Ki > 10000 nM T13201 CNZX07 145953044 Ki > 10000 nM T13201 C5C9RI 145953173 Ki = 3771.1 nM T13201 C1KQ3D 145953178 Ki = 336.8 nM T13201 CQM0J4 145953285 Ki = 57.2 nM T13201 C5DJY9 145953324 Ki = 1471.2 nM T13201 CK5C4D 145953364 Ki = 613 nM T13201 CZO1Y8 145953466 Ki = 65.2 nM T13201 CFW94A 145953493 Ki = 686.3 nM T13201 CX37LN 145953547 Ki = 417 nM T13201 C80OQZ 145953572 Ki = 86.8 nM T13201 C7Q4IN 145953662 Ki > 10000 nM T13201 C36ENH 145953837 Ki = 73.5 nM T13201 CH9N6D 145954010 Ki = 977.1 nM T13201 CVNE29 145954045 Ki = 926.8 nM T13201 C7GIQ5 145954093 Ki > 10000 nM T13201 CD52IH 145954185 Ki = 453 nM T13201 CM4U3B 145954289 Ki = 66.6 nM T13201 C8R2HO 145954507 Ki = 258 nM T13201 C7LZ1G 145954524 Ki = 2847.2 nM T13201 C67HYG 145954632 Ki > 10000 nM T13201 CZG7I4 145954697 Ki = 7.9 nM T13201 CC08PM 145954740 Ki = 79.7 nM T13201 C0XO6A 145954770 Ki = 464.3 nM T13201 CTV8L5 145954775 Ki > 10000 nM T13201 CJ37XC 145954792 Ki = 380 nM T13201 CNE86C 145954868 Ki = 9.6 nM T13201 C1LFA9 145954917 Ki = 4365.5 nM T13201 CMZ2Y0 145954932 Ki = 256.2 nM T13201 C0UBV8 145955012 Ki = 33.2 nM T13201 C7QL4I 145955037 Ki = 294.2 nM T13201 C6UGK8 145955158 Ki = 966.3 nM T13201 CM9Y2S 145955268 Ki = 7069 nM T13201 C0UG3K 145955383 Ki = 847.6 nM T13201 CHTR07 145955486 Ki = 55.6 nM T13201 CS6GA9 145955537 Ki = 272.2 nM T13201 C27JZH 145955576 Ki = 61.9 nM T13201 CW90OF 145955720 Ki = 330.3 nM T13201 CI64UX 145955888 Ki > 10000 nM T13201 CB86QZ 145955914 Ki = 671.8 nM T13201 CG7W8R 145955929 Ki = 747.3 nM T13201 CDWF95 145955978 Ki = 272.1 nM T13201 C9DLX6 145955997 Ki > 10000 nM T13201 CMGN62 145956070 Ki = 183.1 nM T13201 CS93JU 145956073 Ki = 85.4 nM T13201 CDJV68 145956076 Ki = 343.4 nM T13201 C5W1UM 145956081 Ki > 10000 nM T13201 CHXP91 145956144 Ki = 35.6 nM T13201 CZK0L8 145956164 Ki = 9.3 nM T13201 CY1AD2 145956169 Ki = 3.9 nM T13201 CD3LK5 145956229 Ki = 552.6 nM T13201 C89HDL 145956309 Ki = 73.5 nM T13201 CYJ3N0 145956346 Ki = 256.8 nM T13201 C2KV9S 145956347 Ki = 428.7 nM T13201 CQJO72 145956348 Ki > 10000 nM T13201 CGY39T 145956363 Ki = 39.1 nM T13201 CEL63H 145956491 Ki = 6.1 nM T13201 CAPD95 145956503 Ki > 10000 nM T13201 C4LH5W 145956563 Ki = 88.9 nM T13201 CRYP47 145956664 Ki > 10000 nM T13201 CE39IU 145956732 Ki > 10000 nM T13201 CYH7O8 145956770 Ki > 10000 nM T13201 CWPZ94 145956803 Ki = 93.3 nM T13201 CRUI17 145956819 Ki = 74.5 nM T13201 C6I1XE 145956976 Ki = 234.3 nM T13201 C7K2DA 145957040 Ki = 317.9 nM T13201 C7X6NA 145957099 Ki = 147.6 nM T13201 CEF41D 145957103 Ki = 567.6 nM T13201 CAMD59 145957136 Ki = 95.6 nM T13201 C94GRZ 145957236 Ki = 633.4 nM T13201 CED18K 145957307 Ki = 1565.7 nM T13201 CC70NV 145957377 Ki = 385 nM T13201 CKOX92 145957394 Ki = 536.1 nM T13201 C17FUI 145957430 Ki = 42.5 nM T13201 CN5TM2 145957461 Ki = 707 nM T13201 C4S7BR 145957546 Ki = 941.9 nM T13201 C98PXC 145957555 Ki = 2141 nM T13201 CL28OB 145957582 Ki > 10000 nM T13201 CP4TF7 145957664 Ki = 666.6 nM T13201 CI5B9M 145957665 Ki > 10000 nM T13201 C6HG7S 145957711 Ki = 517.5 nM T13201 CE4O0N 145957959 Ki = 21.8 nM T13201 CXFV43 145958041 Ki = 410.9 nM T13201 C3LZ9J 145958059 Ki = 514 nM T13201 C6JL8X 145958066 Ki = 733.3 nM T13201 CM07ZF 145958200 Ki = 226.1 nM T13201 CQO8H5 145958250 Ki = 45.8 nM T13201 CF07KV 145958447 Ki = 69.8 nM T13201 C5URQ2 145958565 Ki = 186 nM T13201 CC32ZJ 145958632 Ki = 750.8 nM T13201 C0PRJ7 145958803 Ki = 53.9 nM T13201 C14UQR 145958824 Ki > 10000 nM T13201 C2MCO8 145958917 Ki > 10000 nM T13201 C0F9NS 145958940 Ki = 915.7 nM T13201 C52CMJ 145958993 Ki = 98 nM T13201 CUBA42 145958994 Ki = 30.1 nM T13201 CXVC18 145959110 Ki = 216.3 nM T13201 CNP7C0 145959116 Ki = 429 nM T13201 CU8J0M 145959118 Ki = 953.7 nM T13201 C1HML4 145959374 Ki = 568.6 nM T13201 C37CVT 145959395 Ki > 10000 nM T13201 C0LC9M 145959407 Ki = 9840.2 nM T13201 CGK4O1 145959409 Ki = 905.6 nM T13201 CM5OK6 145959413 Ki = 218.9 nM T13201 CWNS89 145959524 Ki = 261.7 nM T13201 C7J6MA 145959539 Ki > 10000 nM T13201 CJMU23 145959635 Ki = 42.4 nM T13201 CPL41Z 145959905 Ki = 73.2 nM T13201 CK8DX1 145959911 Ki > 10000 nM T13201 CGZ1K8 145959957 Ki = 881.1 nM T13201 C29YFS 145959974 Ki = 145.6 nM T13201 CL0NM5 145960039 Ki = 380.2 nM T13201 C9MSK2 145960116 Ki = 52.2 nM T13201 CH2K1A 145960207 Ki = 2273.7 nM T13201 C2SI5J 145960220 Ki = 531.2 nM T13201 CB49ZJ 145960257 Ki > 10000 nM T13201 C6JND4 145960287 Ki = 8.4 nM T13201 C3JTG4 145960436 Ki = 6776 nM T13201 C89GHI 145960779 Ki = 542.6 nM T13201 CVMF36 145960835 Ki = 8926 nM T13201 CBGV25 145960853 Ki > 10000 nM T13201 CT6U2G 145961010 Ki = 245 nM T13201 CD2X3F 145961133 Ki = 1010.02 nM T13201 CBT85V 145961452 Ki = 8245 nM T13201 C6JG2V 145961631 Ki = 9.7 nM T13201 CDA7G0 145962071 Ki = 44.3 nM T13201 CCYK28 145962259 Ki = 9410 nM T13201 CQV18P 145962416 Ki = 8404 nM T13201 C14OZY 145962693 Ki = 2.9 nM T13201 C34BRN 145962803 Ki = 8952 nM T13201 C36LCF 145962935 Ki = 7016.1 nM T13201 CZ9PL4 145963030 Ki = 3872 nM T13201 CGY68S 145963294 Ki = 9376 nM T13201 CJU15K 145963586 Ki > 10000 nM T13201 CVL39I 145963679 Ki > 10000 nM T13201 CUZ3A5 145963719 Ki > 10000 nM T13201 C5VI0K 145964063 Ki = 44.1 nM T13201 CM71JT 145964104 Ki > 10000 nM T13201 CGTA80 145964130 Ki = 242.7 nM T13201 C9DE8Y 145964275 Ki = 32.7 nM T13201 C4C9IE 145964340 Ki = 267.9 nM T13201 CK21BE 145964400 Ki = 769.7 nM T13201 CAPU84 145964558 Ki = 20.9 nM T13201 C6FE1K 145964671 Ki = 267.4 nM T13201 CTC21S 145964779 Ki = 483.8 nM T13201 C3F4IS 145965133 Ki = 513.7 nM T13201 CGR16W 145965551 Ki = 6450 nM T13201 C6RZT2 145965743 Ki = 923.9 nM T13201 CWHV36 145965762 Ki = 620 nM T13201 CINP09 145966173 Ki = 881.1 nM T13201 C2G8VU 145966250 Ki = 152.3 nM T13201 C5X7FM 145966343 Ki = 856.4 nM T13201 CCDI76 145966475 Ki = 59.4 nM T13201 CMF72D 145966553 Ki > 10000 nM T13201 CQ64RX 145966558 Ki = 4.9 nM T13201 CJ4D0R 145967030 Ki = 233.8 nM T13201 C7SUX3 145967040 Ki = 63.4 nM T13201 C7HZ6V 145967049 Ki = 2290.4 nM T13201 CP8Q9U 145967308 Ki = 4243.7 nM T13201 CFY3M6 145968026 Ki = 501.7 nM T13201 CDYR51 145968242 Ki = 341.8 nM T13201 C10PQH 145968245 Ki = 8.3 nM T13201 CKME70 145968701 Ki = 73.8 nM T13201 CX4D2R 145969379 Ki = 44.4 nM T13201 C9R4VB 145971458 Ki = 57.3 nM T13201 CD9I1U 145971467 Ki = 338.3 nM T13201 CZ71HS 145971486 Ki = 51.2 nM T13201 C73WMA 145971736 Ki = 36.5 nM T13201 C9P6UE 145971793 Ki = 718.7 nM T13201 C6DQK4 145972104 Ki = 71.4 nM T13201 CO4V1G 145972192 Ki = 30.6 nM T13201 CYMF38 145972316 Ki = 54.2 nM T13201 CP9H1U 145972366 Ki = 4001.7 nM T13201 CD42QZ 145972397 Ki = 19.4 nM T13201 CZ2LP7 145972551 Ki = 3611.4 nM T13201 COJ6K4 145972603 Ki = 2883.7 nM T13201 CGE23X 145972719 Ki = 4767 nM T13201 CFXW14 145972912 Ki = 421.9 nM T13201 CF5KR4 145972986 Ki = 86.5 nM T13201 C65ZVF 145973004 Ki = 3424.4 nM T13201 CN20BQ 145973308 Ki = 9269.7 nM T13201 C1I8GK 145973355 Ki = 1962.6 nM T13201 C9MZS1 145973465 Ki = 87 nM T13201 C8UAD6 145973595 Ki = 6829.7 nM T13201 C7Y3WO 145973882 Ki = 7.9 nM T13201 C2C1KE 145973952 Ki = 5630.7 nM T13201 CJ15WQ 145974101 Ki = 746.3 nM T13201 C7ZRI0 145974266 Ki = 630.8 nM T13201 CX5U8J 145974401 Ki = 7.1 nM T13201 CJD0I1 145974412 Ki = 5330 nM T13201 C2MF3Y 145974672 Ki = 8.5 nM T13201 C1QZ7F 145974710 Ki = 64.9 nM T13201 CG5SL1 145974949 Ki = 435.3 nM T13201 CVPA83 145974992 Ki = 5.9 nM T13201 CDU4M5 145975077 Ki = 21.3 nM T13201 C3I2WU 145975151 Ki = 68.4 nM T13201 C5U8RK 145975281 Ki = 728.5 nM T13201 C1VJD3 145975355 Ki = 7602 nM T13201 CBL8Y4 145975424 Ki = 93.8 nM T13201 CT16KB 145975591 Ki = 51.7 nM T13201 CPK17Y 145975721 Ki = 5930 nM T13201 CZVK21 145975933 Ki = 79.3 nM T13201 CQ08AT 145976207 Ki = 3.6 nM T13201 CO9M3B 145976300 Ki = 4830 nM T13201 CI9C6U 145976539 Ki = 42.5 nM T13201 CZ7QU1 145976656 Ki = 6 nM T13201 C2BIZ4 145976658 Ki = 872.7 nM T13201 CHI26Q 145976735 Ki = 534.4 nM T13201 CZWC63 145977536 Ki = 375.9 nM T13201 CH3IC0 145977574 Ki = 2881.6 nM T13201 CUEB47 145977814 Ki = 73.3 nM T13201 C81JIQ 145977869 Ki = 132.5 nM T13201 CL7GH8 145977904 Ki = 2662.6 nM T13201 CK9L7E 145977947 Ki > 10000 nM T13201 C69UQY 145978025 Ki = 81.7 nM T13201 C5QSK0 145978140 Ki = 741.4 nM T13201 CO0J6L 145978583 Ki > 10000 nM T13201 CYG69V 145978605 Ki = 8.1 nM T13201 CYWK54 145978673 Ki = 48.4 nM T13201 C2D1TO 145978690 Ki = 884.2 nM T13201 CA32BT 145978780 Ki = 57.6 nM T13201 CXI41R 145978938 Ki = 4920 nM T13201 CM8KP7 145979094 Ki = 5390 nM T13201 C82LKO 145979169 Ki = 6210 nM T13201 CI34JB 145979332 Ki = 1816 nM T13201 CSPH69 145979414 Ki = 919.6 nM T13201 CQDB02 145979430 Ki = 2377.3 nM T13201 CUDO01 145979473 Ki > 10000 nM T13201 COYX31 145979594 Ki = 654.3 nM T13201 CFUC92 145979600 Ki = 41.6 nM T13201 CXDE63 145979618 Ki = 960 nM T13201 C7ZOM8 145979619 Ki = 9070 nM T13201 CIF72X 145979737 Ki > 10000 nM T13201 CMT6G7 145979772 Ki = 822.8 nM T13201 C8YA0B 145979831 Ki = 206 nM T13201 C5S9JX 145979949 Ki = 30.3 nM T13201 C9H6AW 145979979 Ki = 750 nM T13201 CLFJ74 145980146 Ki = 321.8 nM T13201 CD1IJ2 145980204 Ki = 289.1 nM T13201 CS85AP 145980216 Ki = 3370 nM T13201 CWA24U 145980366 Ki = 872.1 nM T13201 CE3DP8 145980765 Ki = 14.6 nM T13201 C85TGI 145980938 Ki = 979.3 nM T13201 C97LPB 145981035 Ki = 843.6 nM T13201 C1RO4L 145981799 Ki = 2900 nM T13201 C15PEL 145982039 Ki = 637.9 nM T13201 C4DNF7 145982126 Ki = 991.9 nM T13201 C7N6RT 145982437 Ki = 344.5 nM T13201 C2O8PK 145982576 Ki = 272.9 nM T13201 CK8MY4 145982622 Ki = 72.1 nM T13201 CX6Y5G 145982786 Ki = 395 nM T13201 C7M0HW 145982836 Ki = 68 nM T13201 C34LIQ 145982969 Ki = 479.2 nM T13201 CH3EF7 145983056 Ki = 4715.1 nM T13201 CN7G5J 145983107 Ki = 881.2 nM T13201 C90VNX 145983131 Ki = 916.1 nM T13201 C9S0WG 145983404 Ki = 2061.1 nM T13201 CWUJ59 145983568 Ki = 87.1 nM T13201 CB5G4W 145983664 Ki = 8368.4 nM T13201 CF26VG 145983797 Ki = 477.6 nM T13201 C5SLN9 145983850 Ki = 79.7 nM T13201 CI52KO 145983856 Ki = 322.1 nM T13201 C3J5NQ 145983899 Ki = 899.7 nM T13201 C8PM9Y 145984067 Ki = 194.9 nM T13201 CA6I9T 145984095 Ki = 173.8 nM T13201 CEA52W 145984222 Ki = 203.2 nM T13201 CO9P3M 145984354 Ki = 91 nM T13201 C49ALP 145984517 Ki = 655.7 nM T13201 C8C0AB 145984626 Ki = 9467.2 nM T13201 CLDZ58 145984801 Ki = 377.9 nM T13201 C05FCU 145984802 Ki = 71.2 nM T13201 C7N6ZB 145984855 Ki = 613.9 nM T13201 C4FBS2 145985005 Ki = 7616.1 nM T13201 CZ8NA9 145985353 Ki = 554.3 nM T13201 C8Y1UT 145985534 Ki = 53.2 nM T13201 CF16KP 145985651 Ki = 539.7 nM T13201 CJEG52 145985679 Ki = 79.7 nM T13201 CN1WK4 145985761 Ki = 76 nM T13201 CIT98E 145985912 Ki = 232.1 nM T13201 C8VIF2 145985922 Ki = 87.4 nM T13201 CX0YW6 145985969 Ki = 95.2 nM T13201 C3E0RD 145986123 Ki = 88.4 nM T13201 CF7CH8 145986297 Ki = 90.5 nM T13201 CTZ71U 145986436 Ki = 5990 nM T13201 CIDO62 145986509 Ki = 8330 nM T13201 CK05FT 145986641 Ki = 9290 nM T13201 CN56XE 145986933 Ki = 8164.3 nM T13201 CG6CU5 145987209 Ki = 409.3 nM T13201 CT01AM 145987366 Ki > 50000 nM T13201 C9UBE8 145987408 Ki = 7.1 nM T13201 CZPA17 145987454 Ki = 9489.9 nM T13201 CI9F3V 145987533 Ki = 900.9 nM T13201 C65QOW 145987697 Ki = 33.5 nM T13201 CQF4O8 145987804 Ki = 671.8 nM T13201 CBF3V2 145987828 Ki = 665.6 nM T13201 C0LVN9 145987839 Ki = 3549.5 nM T13201 C6RMF1 145987996 Ki = 47.7 nM T13201 C8XDH5 145988129 Ki > 50000 nM T13201 C89RFU 145988368 Ki = 135.2 nM T13201 CJ1P5W 145988462 Ki > 10000 nM T13201 CXA6F3 145988572 Ki = 44.2 nM T13201 CO3N6M 145988784 Ki = 551.8 nM T13201 CPZN93 145988792 Ki = 1485.6 nM T13201 CZW72V 145988876 Ki = 354 nM T13201 C1LV0U 145988936 Ki > 10000 nM T13201 C39ZMI 145988963 Ki = 323.1 nM T13201 C7AUF1 145989028 Ki = 2262.9 nM T13201 C6BKP8 145989063 Ki = 4790 nM T13201 C35VEG 145989087 Ki = 3460 nM T13201 C6DN9E 145989219 Ki = 490 nM T13201 COZM89 145989422 Ki = 1380 nM T13201 CJH51I 145989433 Ki = 8020 nM T13201 C9RVK0 145989853 Ki > 10000 nM T13201 CYJ79A 145989992 Ki = 8.2 nM T13201 CA8K2J 145990039 Ki = 1832.6 nM T13201 C8XD2V 145990044 Ki > 50000 nM T13201 CLQ12A 145990129 Ki = 739 nM T13201 CHMR39 145990191 Ki = 7101.7 nM T13201 CYOD69 145990290 Ki = 7862 nM T13201 CZB2X3 145990392 Ki = 9638.6 nM T13201 CB63XC 145990519 Ki > 10000 nM T13201 CJQ73W 145990589 Ki = 1864.2 nM T13201 C2WTN6 145990640 Ki = 2335.2 nM T13201 CM6SA4 145990881 Ki = 825.3 nM T13201 CIA37P 145991377 Ki = 377.1 nM T13201 CWH89P 145991839 Ki = 2493 nM T13201 C3QXL4 145991981 Ki = 5503.9 nM T13201 C9F8TL 145992666 Ki = 15.8 nM T13201 C58FGU 145992776 Ki > 50000 nM T13201 C7RYJ4 145992796 Ki = 5795.9 nM T13201 CE34YK 145992956 Ki = 4105.9 nM T13201 CH48GI 145992962 Ki = 1434 nM T13201 CO42RK 145992983 Ki = 896.3 nM T13201 C8IE2X 145993014 Ki = 3289.5 nM T13201 CDC84X 145993019 Ki = 2476.5 nM T13201 C7OZD6 145993265 Ki = 42.2 nM T13201 CE0HY6 145993300 Ki = 309.3 nM T13201 CS40WA 145993323 Ki = 414.1 nM T13201 CMS86X 145993352 Ki = 5670 nM T13201 CB12JK 145993432 Ki = 345.8 nM T13201 CZSC36 145993499 Ki = 720.7 nM T13201 CEC07M 145993642 Ki = 8200 nM T13201 CK3YT9 145993866 Ki = 935 nM T13201 CIDP76 145994238 Ki = 2079.8 nM T13201 C48CZD 146160385 Ki = 196.9 nM T13201 C2SG4L 146833326 Ki > 10000 nM T13201 C6FD2N 147348395 Ki = 1894 nM T13201 CGMX98 155510724 Ki = 34.6 nM T13201 C06MEW 155510831 Ki = 263.9 nM T13201 C3QJI5 155510851 Ki = 84.1 nM T13201 CY5T1K 155510897 Ki > 10000 nM T13201 C1PG9M 155511036 Ki = 83.9 nM T13201 CN6DW9 155511075 Ki = 779.7 nM T13201 C2PXC3 155511133 Ki = 816.7 nM T13201 C1A5OB 155511232 Ki = 240.4 nM T13201 C30ADE 155511364 Ki > 10000 nM T13201 C1D8JF 155511459 Ki > 10000 nM T13201 C6QNX5 155511723 Ki = 891 nM T13201 C03BJU 155511800 Ki = 29000 nM T13201 CJA94W 155512108 Ki = 36.5 nM T13201 CMCL94 155512138 Ki = 3267.4 nM T13201 CE59ZG 155512211 Ki = 209.8 nM T13201 CI40CL 155512225 Ki = 311.3 nM T13201 C1ZPW3 155512418 Ki = 378.6 nM T13201 CQC04P 155512706 Ki = 4161 nM T13201 C7J0HP 155512942 Ki > 100000 nM T13201 C51PHM 155512962 Ki > 10000 nM T13201 CN53ED 155512974 Ki > 100000 nM T13201 CVSG61 155513076 Ki = 676.1 nM T13201 C21CAW 155513169 Ki = 89.4 nM T13201 CW1DP7 155513481 Ki = 1137.1 nM T13201 C7QT4V 155513609 Ki > 10000 nM T13201 CX2UJ9 155514131 Ki = 58300 nM T13201 CZ5W1M 155514230 Ki = 703.7 nM T13201 CV7WR4 155514243 Ki > 10000 nM T13201 C67VGD 155514389 Ki = 82.8 nM T13201 CM5J3L 155514471 Ki = 285.5 nM T13201 CDM78Q 155514660 Ki = 256.4 nM T13201 C7W9NI 155514825 Ki = 896 nM T13201 CU9H2A 155514935 Ki = 368.2 nM T13201 CMQV46 155514970 Ki = 817.1 nM T13201 CCQB03 155515285 Ki = 82.1 nM T13201 CW08ZX 155515305 Ki = 24800 nM T13201 C5IPM8 155515308 Ki > 10000 nM T13201 C46UNX 155515514 Ki = 175.4 nM T13201 C6DG3E 155515525 Ki > 100000 nM T13201 C7MER6 155515557 Ki = 9400 nM T13201 C7UQ3J 155515746 Ki = 741 nM T13201 CT2ZB0 155515980 Ki = 6.6 nM T13201 C74SEH 155516204 Ki > 100000 nM T13201 CM9F7H 155516281 Ki = 4025 nM T13201 CZN16J 155516304 Ki = 941.1 nM T13201 CLNT85 155516404 Ki = 895 nM T13201 COP4Q6 155516517 Ki = 470 nM T13201 C9LWV6 155516550 Ki = 2.8 nM T13201 C7IR3P 155516553 Ki = 45900 nM T13201 CBV6D3 155516701 Ki = 357.4 nM T13201 CP0NH3 155516885 Ki > 10000 nM T13201 C2E0ZF 155517026 Ki = 729.9 nM T13201 CAG9L4 155517430 Ki = 2774 nM T13201 C3OW4N 155517544 Ki = 669 nM T13201 CW18JG 155517622 Ki = 722.9 nM T13201 C2H3JR 155517687 Ki > 100000 nM T13201 CQI20B 155517798 Ki = 69700 nM T13201 CRP2A6 155517861 Ki = 558.2 nM T13201 CWP3G6 155517862 Ki > 10000 nM T13201 CHA2R1 155517933 Ki = 302.7 nM T13201 CF07ZS 155517996 Ki = 88.2 nM T13201 C0O5CN 155518098 Ki > 10000 nM T13201 CUN49T 155518138 Ki = 306.9 nM T13201 C92QDE 155518180 Ki = 2035.7 nM T13201 C1VNX3 155518220 Ki = 971.1 nM T13201 CP0U8D 155518225 Ki > 50000 nM T13201 CEH62Y 155518447 Ki = 517.7 nM T13201 CP7UI1 155518510 Ki = 307.8 nM T13201 CM7DQ6 155518807 Ki = 1418.8 nM T13201 CHI59Y 155518875 Ki > 100000 nM T13201 CL92UI 155519026 Ki = 1458.2 nM T13201 C5TO4Q 155519047 Ki > 100000 nM T13201 CRF95N 155519064 Ki = 5312.5 nM T13201 CN8RC2 155519138 Ki = 566 nM T13201 CK21TJ 155519240 Ki = 2546.8 nM T13201 C8MYG2 155519248 Ki = 415.3 nM T13201 CO6D1Y 155519288 Ki = 726.7 nM T13201 CC47MV 155519432 Ki = 479.4 nM T13201 CT56OD 155519473 Ki = 110.6 nM T13201 CI18TP 155519626 Ki > 10000 nM T13201 CO4V0B 155519627 Ki = 68.7 nM T13201 CP4IL9 155519983 Ki = 100.8 nM T13201 CIV68R 155520019 Ki = 397.5 nM T13201 C5PN0D 155520029 Ki > 10000 nM T13201 CP49HE 155520274 Ki = 62.3 nM T13201 C4Z8MX 155520314 Ki = 381.6 nM T13201 C5JCL6 155520507 Ki > 10000 nM T13201 CG4VJ8 155520652 Ki = 59.3 nM T13201 C8E0SN 155520671 Ki = 44000 nM T13201 CE8QY5 155520792 Ki = 716.9 nM T13201 C4LPA1 155520806 Ki = 750.6 nM T13201 C80OQU 155520908 Ki = 8850 nM T13201 CQ0OR1 155520930 Ki > 10000 nM T13201 C9Z1FL 155521038 Ki > 10000 nM T13201 C2J1YG 155521041 Ki = 1705.9 nM T13201 C2PR8W 155521294 Ki = 779.4 nM T13201 CN2X1Q 155521353 Ki = 81.9 nM T13201 CCGT71 155521462 Ki = 15.3 nM T13201 CB54YX 155521489 Ki = 152.9 nM T13201 CF7HE1 155521700 Ki = 2125 nM T13201 CRQ4L3 155521766 Ki = 8174.1 nM T13201 CZ7WI8 155521830 Ki = 52.7 nM T13201 CNP87G 155521876 Ki = 9403.9 nM T13201 CR49AJ 155521885 Ki = 100.5 nM T13201 C4IYX7 155521930 Ki = 724.3 nM T13201 C2Q7BG 155522085 Ki = 1782.5 nM T13201 C0A4EO 155522100 Ki = 597.5 nM T13201 CSN4C2 155522321 Ki = 2244.1 nM T13201 C70NUX 155522372 Ki = 641.3 nM T13201 C8K9OI 155522618 Ki = 8.1 nM T13201 C6AWP0 155522679 Ki = 495.5 nM T13201 CDN9Z5 155522816 Ki = 99 nM T13201 C0Z3QT 155522883 Ki = 5841.5 nM T13201 CJ49ZN 155522995 Ki = 3518.6 nM T13201 CM3H1N 155523109 Ki = 256.6 nM T13201 CA9F2I 155523252 Ki = 108.7 nM T13201 C3HGK6 155523328 Ki = 817.9 nM T13201 C6YZM3 155523403 Ki > 100 nM T13201 C9Q2WR 155523406 Ki = 591.3 nM T13201 CWJ7R5 155523492 Ki = 1.5 nM T13201 CU2N9J 155523547 Ki = 666.5 nM T13201 CIF91M 155523572 Ki = 64.9 nM T13201 C9LF7B 155523634 Ki > 100000 nM T13201 C4U8XN 155523810 Ki = 1413.2 nM T13201 CWD9Y1 155523853 Ki = 347.3 nM T13201 C3MX7F 155523857 Ki = 151.1 nM T13201 C0MZ5G 155524206 Ki = 88.2 nM T13201 C6KCG7 155524248 Ki = 43.1 nM T13201 CSC58M 155524279 Ki > 10000 nM T13201 CK86ZT 155524367 Ki = 3818.1 nM T13201 CK80AQ 155524610 Ki = 939.5 nM T13201 C9PV5X 155524649 Ki = 44500 nM T13201 CS21YC 155524712 Ki = 351.7 nM T13201 CDO4X2 155524724 Ki = 771.4 nM T13201 C3DM5L 155524759 Ki > 10000 nM T13201 C5J8AS 155524785 Ki = 4829.7 nM T13201 CS0WP1 155524852 Ki = 3750 nM T13201 C70ZPH 155524915 Ki = 49.1 nM T13201 C8M1KI 155525036 Ki = 648.5 nM T13201 CV6N0C 155525231 Ki = 507.4 nM T13201 CHT29F 155525313 Ki = 829.6 nM T13201 CA02GS 155526086 Ki = 5093 nM T13201 C4R1OT 155526288 Ki > 50000 nM T13201 CGC8Y0 155526420 Ki > 10000 nM T13201 CKT14B 155526554 Ki > 10000 nM T13201 C0XZD3 155526695 Ki = 8450 nM T13201 CWGS97 155526825 Ki = 929 nM T13201 CGV91K 155527018 Ki = 403.3 nM T13201 CCL7V8 155527060 Ki = 1317.4 nM T13201 CNVX86 155527078 Ki = 697.7 nM T13201 CAMY18 155527145 Ki = 41.1 nM T13201 CG8JZ9 155527153 Ki = 1536.5 nM T13201 C8K3OI 155527167 Ki = 406.9 nM T13201 C1LDV0 155527209 Ki = 987.7 nM T13201 C1I5PO 155527240 Ki = 3840 nM T13201 CK8XN6 155527284 Ki > 10000 nM T13201 C4N7OY 155527400 Ki = 1163.3 nM T13201 CJ3K9W 155527428 Ki = 898 nM T13201 C4A5BC 155527483 Ki = 4752.2 nM T13201 C7YW9E 155527622 Ki = 6630 nM T13201 CDE96Y 155527673 Ki = 86.1 nM T13201 C65FOA 155527703 Ki = 5842.3 nM T13201 C07LVI 155527781 Ki = 96.2 nM T13201 CPAH30 155527788 Ki = 1955.2 nM T13201 C5XC7V 155527967 Ki > 10000 nM T13201 CDN05K 155527975 Ki = 50.8 nM T13201 C0RJ2M 155528294 Ki = 824.6 nM T13201 CN9G0E 155528332 Ki > 50000 nM T13201 C4IML7 155528345 Ki = 864.2 nM T13201 CLF2V0 155528496 Ki = 501.7 nM T13201 C38SKR 155528605 Ki = 227.1 nM T13201 CB08MU 155528753 Ki = 33500 nM T13201 C2LF1H 155528761 Ki = 105.1 nM T13201 C5X0CS 155528825 Ki > 100000 nM T13201 CN27OU 155528858 Ki = 4545.1 nM T13201 C7DCG0 155529026 Ki = 691.3 nM T13201 CECZ45 155529036 Ki = 4601 nM T13201 C1T2EA 155529101 Ki = 476.5 nM T13201 CWEQ38 155529122 Ki = 192 nM T13201 C52QUD 155529352 Ki = 30.2 nM T13201 C8DN2F 155529373 Ki = 7797 nM T13201 CG94RZ 155529376 Ki = 736.8 nM T13201 C2HUS1 155529422 IC50 = 44.05 nM T13201 C2NY1E 155529877 Ki = 686 nM T13201 C2JV7R 155529885 Ki = 2894 nM T13201 CG3J0Q 155529984 Ki = 618.4 nM T13201 CJ21OD 155530289 Ki > 50000 nM T13201 CW07EO 155530326 Ki = 41.9 nM T13201 CKO2V5 155530358 Ki = 365.4 nM T13201 C7TV5H 155530408 Ki = 54.5 nM T13201 CIGQ50 155530440 Ki = 798.8 nM T13201 C9Y4VC 155530502 Ki = 82.4 nM T13201 CTJ3I7 155530506 Ki = 383.6 nM T13201 C0HQ8E 155530537 Ki = 951.8 nM T13201 CP3UJ0 155530687 Ki = 37.5 nM T13201 C2T0LQ 155530848 Ki = 827 nM T13201 C3GK9H 155530900 Ki = 6936 nM T13201 C2MT3K 155530925 Ki = 3298.5 nM T13201 C8C4BT 155531090 Ki = 454 nM T13201 CICU68 155531183 Ki > 10000 nM T13201 CGN43T 155531186 Ki = 700 nM T13201 CO7P5W 155531268 Ki = 6.5 nM T13201 CLMZ93 155531382 Ki = 242.1 nM T13201 CYBD02 155531537 Ki = 3297 nM T13201 C43LZI 155531630 Ki = 415.8 nM T13201 CC5L6V 155531813 Ki > 2000 nM T13201 CFV23M 155531820 Ki > 100000 nM T13201 CW6TC5 155531936 Ki = 57400 nM T13201 CUM2B8 155532026 Ki > 100000 nM T13201 C83DJY 155532441 Ki > 100000 nM T13201 CASV53 155532466 Ki = 2956.1 nM T13201 CFK8R5 155532512 Ki > 100000 nM T13201 CQ0XM6 155532587 Ki = 935.8 nM T13201 C5H8QF 155532861 Ki = 4042.3 nM T13201 CKY1I8 155533416 Ki = 738.4 nM T13201 CDM2Y1 155533454 Ki = 8.9 nM T13201 C64XYO 155533459 Ki = 5.8 nM T13201 C0BNY7 155533528 Ki = 737.1 nM T13201 CPX2T1 155533590 Ki > 10000 nM T13201 COK37H 155533887 Ki = 6690 nM T13201 CTKI39 155533898 Ki = 7832.9 nM T13201 C0I5XS 155534055 Ki = 60.1 nM T13201 C78ZFI 155534074 Ki = 394.4 nM T13201 CT5NG1 155534179 Ki = 63.6 nM T13201 CPG13Y 155534247 Ki = 94.4 nM T13201 C6UF3R 155534332 Ki = 358 nM T13201 CR2A6J 155534340 Ki > 50000 nM T13201 C14TGQ 155534675 Ki = 437.7 nM T13201 CS0FK9 155534753 Ki = 8.9 nM T13201 CK4TR2 155534861 Ki > 10000 nM T13201 CS5OI9 155534862 Ki = 758.5 nM T13201 CHG10E 155534912 Ki = 481.5 nM T13201 C0QW8K 155535058 Ki = 377.1 nM T13201 CE1I8S 155535343 Ki = 8120 nM T13201 CC7M4N 155535347 Ki > 10000 nM T13201 CVU5P6 155535355 Ki = 80.3 nM T13201 CV0N9I 155535382 Ki > 10000 nM T13201 CKR07J 155535598 Ki > 10000 nM T13201 CNFR72 155535756 Ki = 66600 nM T13201 CFYA23 155535780 Ki = 314.1 nM T13201 CD2O3A 155535852 Ki > 50000 nM T13201 CLJ64Q 155535889 Ki = 67.4 nM T13201 CZPY79 155536184 Ki = 432.1 nM T13201 CF0PC4 155536422 Ki > 10000 nM T13201 CW92OP 155536652 Ki = 2338.4 nM T13201 CB47KF 155536691 Ki = 4638.8 nM T13201 C0EDQ2 155536876 Ki = 513.5 nM T13201 CZ0T6A 155537018 Ki = 2071 nM T13201 COP2R4 155537042 Ki = 350.4 nM T13201 C6T7BQ 155537167 Ki = 3075 nM T13201 C1K9AC 155537404 Ki > 10000 nM T13201 CXQ23T 155537493 Ki > 100000 nM T13201 C4K0MB 155537772 Ki = 530 nM T13201 C0CG6Q 155537790 Ki = 659.7 nM T13201 C47OHJ 155537809 Ki = 231.4 nM T13201 C67ZET 155537843 Ki = 46.9 nM T13201 CYM0A3 155538069 Ki = 101.8 nM T13201 C5RV9W 155538073 Ki = 9.1 nM T13201 COX74J 155538083 Ki = 369.6 nM T13201 C60IZQ 155538189 Ki > 50000 nM T13201 CB2EI4 155538212 Ki = 95.4 nM T13201 C9AP8F 155538224 Ki = 759.4 nM T13201 CB8C4X 155538289 Ki = 54700 nM T13201 C3XSM6 155538611 Ki > 10000 nM T13201 CM6D1H 155538676 Ki > 10000 nM T13201 CHQP36 155539441 Ki = 568.9 nM T13201 CKE72Y 155539552 Ki = 5.4 nM T13201 C94OZU 155539579 Ki > 10000 nM T13201 C9K2TL 155539730 Ki = 2642 nM T13201 CS1G5V 155539783 Ki = 3264 nM T13201 CS1UR7 155539868 Ki = 81.5 nM T13201 C85YWZ 155539989 Ki = 2401 nM T13201 C53TKA 155540088 Ki > 2000 nM T13201 CSAD81 155540401 Ki = 521.3 nM T13201 CZ8FJ3 155540422 Ki = 819.3 nM T13201 CW9B0X 155540441 Ki = 1834.7 nM T13201 C2VAD8 155540596 Ki = 454 nM T13201 C95TBC 155540629 Ki = 37.3 nM T13201 CCO34J 155540665 Ki > 10000 nM T13201 CGNS87 155540756 Ki = 53 nM T13201 CFN03K 155540920 Ki = 384.2 nM T13201 C4H1ZC 155541040 Ki = 2260.1 nM T13201 C3CLU2 155541078 Ki = 569 nM T13201 C7Z6FC 155541724 Ki > 10000 nM T13201 C8RV6T 155541805 Ki = 648.6 nM T13201 CW96ES 155541807 Ki = 564.1 nM T13201 C4MW9Q 155541811 Ki = 91.3 nM T13201 C5F3SJ 155541888 Ki = 2898.4 nM T13201 CX20DK 155541945 Ki = 3212 nM T13201 CZ2CT0 155542259 Ki > 50000 nM T13201 CW61DF 155542555 Ki = 295.6 nM T13201 CA75HO 155542580 Ki = 633.1 nM T13201 CTL8O3 155542606 Ki = 949 nM T13201 C3RC8T 155542635 Ki = 87.4 nM T13201 CT9GZ2 155542660 Ki = 925.7 nM T13201 CDK2W5 155542691 Ki = 748.1 nM T13201 CA76LB 155542698 Ki = 8300 nM T13201 CY3BO6 155542934 Ki = 852.3 nM T13201 C75TVG 155542954 Ki = 8798.6 nM T13201 C2AEH6 155543096 Ki > 50000 nM T13201 CN2SJ7 155543228 Ki = 764.2 nM T13201 C19DJA 155543271 Ki = 82.2 nM T13201 CHKV89 155543295 Ki = 25 nM T13201 CRF64E 155543422 Ki = 266.1 nM T13201 CLF3N5 155543891 Ki = 485.3 nM T13201 CPV20B 155543950 Ki = 3752.5 nM T13201 C08DHT 155544006 Ki > 10000 nM T13201 C30HST 155544165 Ki = 644.7 nM T13201 CN0E1V 155544321 Ki = 681 nM T13201 CS9WR6 155544336 Ki > 2000 nM T13201 C7PC5J 155544382 Ki = 89.7 nM T13201 CSX2H7 155544608 Ki = 3721.8 nM T13201 CI2T8N 155544664 Ki = 51 nM T13201 CRM69J 155544710 Ki = 1607.4 nM T13201 CP27AW 155544846 Ki > 10000 nM T13201 CDXL09 155544901 Ki = 30.7 nM T13201 C0BV1J 155545536 Ki = 805.2 nM T13201 CQV78W 155545657 Ki = 694.9 nM T13201 CB6J9G 155545674 Ki > 10000 nM T13201 CY6SX5 155545800 Ki = 60000 nM T13201 CP2SZ7 155545812 Ki = 8060 nM T13201 C95IJM 155545916 Ki = 1667 nM T13201 CSW62L 155546892 Ki = 21900 nM T13201 CF3UL5 155547275 Ki = 2977.2 nM T13201 CV7OB5 155547342 Ki > 100000 nM T13201 C9E2KH 155547486 Ki = 6567.1 nM T13201 C59MDT 155547507 Ki = 522.7 nM T13201 C83ZIS 155547526 Ki = 494.9 nM T13201 CW19PC 155547551 Ki = 763 nM T13201 C73YLV 155547628 Ki = 67.4 nM T13201 C9FVY6 155547723 Ki = 970.2 nM T13201 C61MSB 155547730 Ki = 46.8 nM T13201 CK5UD3 155547819 Ki = 4083 nM T13201 CP4N3X 155547901 Ki = 24 nM T13201 CU94YA 155548070 Ki > 2000 nM T13201 CCUN29 155548118 Ki = 4142.4 nM T13201 C3IO2B 155548134 Ki > 10000 nM T13201 C3JYG2 155548272 Ki = 1225.3 nM T13201 CQG5F9 155548326 Ki = 1635 nM T13201 C6XBZ3 155548352 Ki = 50.1 nM T13201 CUTY40 155548640 Ki = 607.2 nM T13201 CH2KB7 155548697 Ki = 343.9 nM T13201 CN7S5W 155548866 Ki = 537.1 nM T13201 CDC0F4 155548911 Ki = 102.3 nM T13201 CU1NE7 155549031 Ki = 306.3 nM T13201 CA25QH 155549266 Ki = 441.4 nM T13201 CR79SY 155549354 Ki = 7697 nM T13201 CL2B4T 155549378 Ki = 90.7 nM T13201 C6PY2G 155549478 Ki = 15.3 nM T13201 C2CLU0 155549558 Ki = 494.9 nM T13201 CIG6A7 155549616 Ki = 121 nM T13201 C1JR2F 155549662 Ki > 10000 nM T13201 CF6CW3 155549677 Ki = 522.2 nM T13201 C8NS5F 155549723 Ki = 813 nM T13201 CEZX49 155549753 Ki = 1308.4 nM T13201 C8GZK4 155549788 Ki > 100000 nM T13201 CAYO49 155550021 Ki = 2140.9 nM T13201 C3YN0W 155550099 Ki = 382.2 nM T13201 CZB57Y 155550558 Ki = 97.4 nM T13201 CHO96B 155550610 Ki = 10900 nM T13201 C4O6TN 155550616 Ki = 390.8 nM T13201 CMWQ79 155550618 Ki = 6422.9 nM T13201 C6XPV0 155550626 Ki = 816.3 nM T13201 CB2Q4M 155550927 Ki = 2292 nM T13201 CG0MQ3 155551020 Ki = 89 nM T13201 CTE04H 155551088 Ki = 4133 nM T13201 CPRC19 155551316 Ki = 61.9 nM T13201 C4S0JZ 155551334 Ki = 8345 nM T13201 CL2H8V 155551536 Ki > 100000 nM T13201 CSY39H 155551651 Ki = 800 nM T13201 C69AYQ 155551705 Ki > 100000 nM T13201 COC4Z9 155551784 Ki = 195.1 nM T13201 CZ0T3C 155551786 Ki = 39.3 nM T13201 C3AN2K 155551935 Ki = 2446 nM T13201 CG9PN8 155552113 Ki = 87.3 nM T13201 C7E3UF 155552316 Ki = 80600 nM T13201 C3DHB7 155552411 Ki > 50000 nM T13201 CW8S7L 155552594 Ki = 3285 nM T13201 CN25FV 155552708 Ki = 365 nM T13201 CBQ42J 155552773 Ki = 19800 nM T13201 CFT82G 155552780 Ki = 2496.4 nM T13201 C0OG8P 155553361 Ki = 0.63 nM T13201 CP15VC 155553400 Ki = 8365 nM T13201 C1QJ3H 155553542 Ki = 456.6 nM T13201 C82WXR 155553544 Ki = 5886.8 nM T13201 CQM27S 155553591 Ki = 5095.8 nM T13201 CQ1PE4 155553611 Ki > 100000 nM T13201 C1R7CJ 155553759 Ki = 9.2 nM T13201 C02LSY 155553787 Ki > 10000 nM T13201 C6IMR3 155554140 Ki = 2313.3 nM T13201 CMEP40 155554179 Ki = 317.9 nM T13201 CE57CO 155554263 Ki = 809 nM T13201 C0U8CG 155554286 Ki = 5939.5 nM T13201 C6D9BJ 155554303 Ki > 10000 nM T13201 C3W6RT 155554309 Ki = 6250 nM T13201 CNX5L2 155554533 Ki = 840.9 nM T13201 C5VLU4 155554670 Ki > 10000 nM T13201 CM4I0O 155554763 Ki = 39600 nM T13201 CZU9Y7 155554800 Ki = 75.5 nM T13201 CW5F4A 155554840 Ki = 681.1 nM T13201 C5YA7C 155555084 Ki = 1066 nM T13201 C9W1ET 155555489 Ki > 10000 nM T13201 CJ06PN 155555584 Ki = 173 nM T13201 CV2NZ0 155555718 Ki = 415.4 nM T13201 CUY2C6 155555751 Ki = 7.9 nM T13201 CA7UK2 155555803 Ki = 97.3 nM T13201 CXNZ49 155555817 Ki = 8.9 nM T13201 CX4P1W 155555874 Ki = 2481 nM T13201 CWB82E 155555878 Ki = 490.8 nM T13201 CKIR52 155556062 Ki = 96.8 nM T13201 C84MNE 155556163 Ki = 312.6 nM T13201 C5PZF2 155556257 Ki = 1030.5 nM T13201 CM60WT 155556386 Ki = 1676.8 nM T13201 CD4K6H 155556521 Ki = 6.3 nM T13201 CVR2X5 155556659 Ki > 100000 nM T13201 CGZ58Y 155556761 Ki = 89.7 nM T13201 C2Q3UO 155556889 Ki = 3265.4 nM T13201 CYZ3K0 155556908 Ki = 702.7 nM T13201 CG8L0O 155557058 Ki > 10000 nM T13201 CHKA19 155557282 Ki = 227.4 nM T13201 CJF9O7 155557300 Ki = 52500 nM T13201 C87GRH 155557329 Ki = 3131.7 nM T13201 CRK5I0 155557428 Ki = 1778 nM T13201 C40MOH 155557452 Ki = 7.3 nM T13201 C1RMC6 155557757 Ki > 10000 nM T13201 CNX9J2 155557875 Ki = 8253.1 nM T13201 CM6NU0 155557925 Ki = 442.3 nM T13201 CWK35T 155557969 Ki = 334.6 nM T13201 CQI5Z4 155558076 Ki > 10000 nM T13201 CK8GH2 155558119 Ki = 48 nM T13201 CME2Z4 155558216 Ki = 46.5 nM T13201 C70WSB 155558230 Ki > 10000 nM T13201 CQ2ML6 155558561 Ki > 50000 nM T13201 CK1RO0 155558641 Ki = 16.2 nM T13201 CH1Z2S 155558695 Ki = 7000 nM T13201 C4V2PS 155558747 Ki = 5225.3 nM T13201 C6QXP8 155558748 Ki > 50000 nM T13201 CZ7C0S 155558990 Ki = 242.1 nM T13201 CI2XS3 155559081 Ki = 295.2 nM T13201 C6CY3G 155559512 Ki = 95.1 nM T13201 CNT0F5 155559682 Ki > 10000 nM T13201 CK7H8I 155559761 Ki = 755 nM T13201 C3Y7WJ 155560101 Ki = 67400 nM T13201 CZ2A7O 155560148 Ki = 1024.1 nM T13201 CB2X0V 155560428 Ki > 10000 nM T13201 CB5S8V 155560635 Ki = 122.1 nM T13201 COC45S 155560702 Ki = 6147.9 nM T13201 CY1TF7 155560798 Ki = 88.2 nM T13201 C0U1NP 155560951 Ki = 6.5 nM T13201 CFY9A2 155561027 Ki = 276 nM T13201 CP3H0R 155561119 Ki > 100000 nM T13201 C3FG8W 155561198 Ki = 7300 nM T13201 CSK5X2 155561354 Ki > 10000 nM T13201 C2SZM0 155561361 Ki = 188.4 nM T13201 CAP5I4 155561568 Ki = 2741.9 nM T13201 CU03LF 155561751 Ki = 9590.6 nM T13201 CY9N4P 155561775 Ki > 50000 nM T13201 CU1JV7 155561839 Ki = 7981.2 nM T13201 CJ5Y6X 155561851 Ki > 10000 nM T13201 CXE2R9 155561928 Ki = 188.1 nM T13201 C5W7MQ 155562360 Ki = 3408.1 nM T13201 CG43PS 155562766 Ki = 72.6 nM T13201 C2FW8S 155562815 Ki = 129.8 nM T13201 CJ74ND 155563017 Ki = 28.7 nM T13201 C1J3UH 155563153 Ki > 100000 nM T13201 C7A8EX 155563186 Ki = 5890.7 nM T13201 C9SH6R 155563203 Ki > 100000 nM T13201 C6KD7C 155563215 Ki = 512.9 nM T13201 CP85AZ 155563623 Ki = 886.7 nM T13201 C89MTB 155563810 Ki = 8981 nM T13201 C0GU6P 155563888 Ki > 10000 nM T13201 CQ40DU 155563908 Ki = 886 nM T13201 C2XB6V 155564028 Ki > 10000 nM T13201 CF7XH2 155564101 Ki = 458.7 nM T13201 CGY32K 155564210 Ki = 8292.5 nM T13201 CY9M4F 155564463 Ki > 50000 nM T13201 C97TMY 155564559 Ki = 4130 nM T13201 C1K0LR 155564617 Ki = 793.4 nM T13201 C07GFY 155564664 Ki = 6092 nM T13201 CY9IW2 155564942 Ki = 292.3 nM T13201 CNV35X 155565135 Ki = 1539.2 nM T13201 C0XO6Z 155565139 Ki = 7331 nM T13201 C0E4QV 155565149 Ki = 44.1 nM T13201 C5XV7O 155565283 Ki = 8.3 nM T13201 CNL8B7 155565372 Ki = 6348.3 nM T13201 CI5MV1 155565395 Ki = 2071.3 nM T13201 CJ7I6Z 155565419 Ki = 670.7 nM T13201 CDF5E6 155565628 Ki = 6178 nM T13201 C0COK6 155565635 Ki = 4953.5 nM T13201 CT9Z5H 155565773 Ki > 50000 nM T13201 CW3N9Z 155566095 Ki > 10000 nM T13201 CD6Z0B 155566206 Ki = 101.4 nM T13201 COA9F8 155566222 Ki = 71300 nM T13201 CCW3L7 155566305 Ki > 50000 nM T13201 CJQP47 155566378 Ki = 960.2 nM T13201 C5QAM3 155566668 Ki = 459.3 nM T13201 CBV30Y 155566701 Ki = 2381.9 nM T13201 CA6JT2 155566730 Ki = 18 nM T13201 CI8U3W 155566755 Ki = 720.3 nM T13201 CA63FB 155566994 Ki = 939.4 nM T13201 CK80EL 155567119 Ki = 4697 nM T13201 C4TZ8Q 155567475 Ki = 441.7 nM T13201 CK0M8P 155567487 Ki = 676.6 nM T13201 CL1N9Y 155567612 Ki > 100000 nM T13201 C1MHV5 155567738 Ki > 10000 nM T13201 C29EYS 155567759 Ki > 10000 nM T13201 CJ2YC4 155567804 Ki = 9.3 nM T13201 C9DOG1 155567981 Ki = 4963 nM T13201 CZP30I 155567991 Ki = 227.8 nM T13201 CCX06Y 155568045 Ki = 3208.5 nM T13201 CN5OF0 155568108 Ki = 587 nM T13201 C2ZRJ3 155568270 Ki = 172.2 nM T13201 CG82MB 155568274 Ki = 2579.9 nM T13201 CDB8T4 155568445 Ki = 7.7 nM T13201 C94QKZ 155568447 Ki = 2669 nM T13201 C52NQU 155568453 Ki = 7.8 nM T13201 C35XQY 155568474 Ki = 4484.3 nM T13201 C6KR4H 155568759 Ki > 10000 nM T13201 CH5VU6 155568899 Ki = 853.1 nM T13201 C1C2GI 155569076 Ki = 75.5 nM T13201 C83MGT 155569151 Ki = 649 nM T13201 CAUR85 155569555 Ki = 4900 nM T13201 C1A7IN 155569676 Ki = 59.3 nM T13201 D00BMI 25154729 Ki = 7420 nM T13201 D00FGB 11414131 Ki = 7.1 nM T13201 D00GVA 44520904 Ki = 71 nM T13201 D00IAE 11974340 Ki = 4000 nM T13201 D00IKQ 46703766 Ki = 7340 nM T13201 D00IUB 13019 Ki = 131000 nM T13201 D00LFX 20718630 Ki = 15 nM T13201 D00NUK 2837872 Ki = 125 nM T13201 D00RJT 943 Ki = 7000000 nM T13201 D00RNZ 910172 Ki = 26900 nM T13201 D00SXO 2793709 Ki > 10000 nM T13201 D00TRF 44423683 Ki = 490000 nM T13201 D00XIB 11680415 Ki = 8.5 nM T13201 D00XJA 711717 Ki = 59 nM T13201 D00YEF 148885 Ki = 890 nM T13201 D01BUB 94952 Ki = 134000 nM T13201 D01CXM 52949265 Ki > 100000 nM T13201 D01EEM 462919 Ki = 276 nM T13201 D01FOK 52949288 Ki > 100000 nM T13201 D01GNQ 44395086 Ki = 31700000 nM T13201 D01ISX 670786 Ki = 68 nM T13201 D01JTI 11687831 Ki = 1095 nM T13201 D01KKU 5281894 Ki = 3370 nM T13201 D01OTW 46703932 Ki = 11710 nM T13201 D01STY 9861037 Ki = 6000 nM T13201 D01UDU 11287480 Ki = 2800 nM T13201 D01UYI 5281607 Ki = 5420 nM T13201 D01XFH 11851424 Ki = 6100 nM T13201 D01YHK 10932611 Ki = 3300 nM T13201 D02BMV 46907399 Ki = 8320 nM T13201 D02DBP 5054 Ki = 795000 nM T13201 D02DCD 45483280 Ki = 8270 nM T13201 D02JEZ 5281426 Ki > 10000 nM T13201 D02KDH 11160546 Ki = 48300 nM T13201 D02MAK 5705744 Ki > 100000 nM T13201 D02NQK 46703924 Ki = 7620 nM T13201 D02QGI 273 Ki = 13300 nM T13201 D03APP 4386 Ki = 1200 nM T13201 D03DAM 2725651 Ki = 5900 nM T13201 D03KRB 45028567 Ki = 11170 nM T13201 D03LHJ 52946829 Ki > 100000 nM T13201 D03MJM 45273020 IC50 = 129000000 nM T13201 D03NBX 637308 Ki > 50000 nM T13201 D03VUQ 404202 Ki = 80 nM T13201 D03ZMQ 323 Ki = 3100 nM T13201 D04BKU 148886 Ki = 548 nM T13201 D04CVC 4687472 Ki = 8300 nM T13201 D04HQK 394898 Ki = 38 nM T13201 D04JIN 44405179 Ki = 5200 nM T13201 D04LNI 75490 Ki = 92800 nM T13201 D04NSN 169682 Ki = 94.7 nM T13201 D04POB 8482 Ki = 21400 nM T13201 D04PSK 44571848 Ki = 2400 nM T13201 D04RCR 11041016 Ki = 8600 nM T13201 D04SNH 46933593 Ki = 4120 nM T13201 D04VSP 46703768 Ki = 6100 nM T13201 D05BMD 44423684 Ki = 10000 nM T13201 D05DIH 45483180 Ki = 7460 nM T13201 D05EBZ 46703769 Ki = 6640 nM T13201 D05ETN 46703923 Ki = 10320 nM T13201 D05FMD 9447 IC50 = 4070 nM T13201 D05FNN 100606 Ki = 145 nM T13201 D05JAJ 45028568 Ki = 10320 nM T13201 D05NFU 4100860 Ki = 7900 nM T13201 D05QEK 44395692 Ki = 62 nM T13201 D05QOR 5280460 Ki = 10560 nM T13201 D05QUG 45485279 Ki = 31400 nM T13201 D05RAB 45028895 Ki = 3440 nM T13201 D05TLB 11117301 Ki = 3.5 nM T13201 D05VUA 850202 Ki > 100000 nM T13201 D05VVC 44315786 Ki > 10000 nM T13201 D05WQF 637540 Ki = 3100 nM T13201 D05XZM 10081162 Ki = 55 nM T13201 D06ALC 6441498 Ki > 10000 nM T13201 D06DYP 234562 Ki = 66 nM T13201 D06GPL 44405177 Ki = 952 nM T13201 D06IOI 901953 Ki = 9090 nM T13201 D06IYU 15569631 Ki = 13 nM T13201 D06JVR 44571849 Ki = 1660 nM T13201 D06KTD 2490720 Ki = 24500 nM T13201 D06MZK 31405 Ki = 274500 nM T13201 D06NDR 44423687 Ki = 10200 nM T13201 D06ORV 65389 Ki = 11400 nM T13201 D06SME 46871781 IC50 = 210 nM T13201 D06SZG 44315523 Ki > 10000 nM T13201 D06TPF 1057 Ki = 7410 nM T13201 D06WZG 50925425 Ki > 100000 nM T13201 D06XNT 4119643 Ki = 75 nM T13201 D06XVV 64048 Ki > 500000 nM T13201 D06ZMH 2812287 Ki = 1500 nM T13201 D06ZOM 15569045 Ki > 10000 nM T13201 D07AGM 14612854 Ki = 25000 nM T13201 D07AUN 969280 Ki = 1040 nM T13201 D07CBA 44391592 Ki = 16450 nM T13201 D07CQI 42546 Ki = 35800 nM T13201 D07CYN 20347846 Ki = 33 nM T13201 D07IHP 44391650 Ki = 79 nM T13201 D07IRQ 7478 Ki = 9060 nM T13201 D07LYW 11537386 Ki = 4130 nM T13201 D07MQB 10903168 Ki = 3700 nM T13201 D07MTM 403 Ki = 159000 nM T13201 D07OMY 44574267 Ki = 48 nM T13201 D07PNA 11660633 Ki = 5330 nM T13201 D07QIU 625902 Ki > 50000 nM T13201 D07QJJ 289 Ki = 4003000 nM T13201 D07SIA 78318 Ki = 1250 nM T13201 D07TAJ 914298 Ki = 224000 nM T13201 D07VXX 16721024 Ki = 435000 nM T13201 D07YDN 5281654 Ki > 10000 nM T13201 D07YSQ 10385283 Ki = 40 nM T13201 D07ZXR 44391576 Ki = 1350 nM T13201 D08AIJ 440735 Ki > 10000 nM T13201 D08AOA 11543564 Ki = 3440 nM T13201 D08BFU 5282102 Ki > 10000 nM T13201 D08JCC 46703770 Ki = 9160 nM T13201 D08JNO 52943193 Ki > 100000 nM T13201 D08XQI 9395 IC50 = 338 nM T13201 D09CSP 3161908 Ki = 6690 nM T13201 D09CXX 16122590 Ki = 4050 nM T13201 D09FQL 16756780 Ki = 368000 nM T13201 D09JHA 33558 Ki = 1200 nM T13201 D09JPC 16402 Ki = 12600 nM T13201 D09LUD 4229592 Ki = 430 nM T13201 D09LWR 3433937 Ki = 60 nM T13201 D09OSN 151253 Ki = 3700 nM T13201 D09PWX 8739 Ki = 109 nM T13201 D09QHC 7370 Ki = 12360 nM T13201 D09TES 44395768 Ki = 89 nM T13201 D09TKG 25044690 Ki = 8860 nM T13201 D09USO 5277466 IC50 > 10000 nM T13201 D09WSJ 19772348 Ki = 530 nM T13201 D09WVV 8111 Ki = 415000 nM T13201 D09ZUN 10269 Ki = 63700 nM T13201 D0A0RT 11602828 Ki = 37900 nM T13201 D0A0YX 5143 Ki > 10000 nM T13201 D0A1CM 5281855 Ki = 2320 nM T13201 D0A3JR 3051968 Ki = 61 nM T13201 D0A4HS 201262 Ki = 10900 nM T13201 D0A4TC 446504 Ki = 281000 nM T13201 D0A6HS 6852129 Ki = 55 nM T13201 D0A8HW 44395685 Ki = 36 nM T13201 D0AU0M 637542 Ki = 1070 nM T13201 D0B0SD 104745 Ki = 1010000 nM T13201 D0B4IN 375084 Ki = 4350 nM T13201 D0B5GC 11349 Ki = 5100 nM T13201 D0BR1D 13443185 IC50 = 7640 nM T13201 D0C3SL 67185 Ki = 37500 nM T13201 D0C4QB 44395769 Ki = 43 nM T13201 D0C7LR 313 Ki = 6000000 nM T13201 D0C8ZY 2734375 Ki = 6500 nM T13201 D0C9ZY 11804953 Ki = 55600 nM T13201 D0CM3O 446142 Ki = 7700 nM T13201 D0D0BO 180598 Ki = 9.6 nM T13201 D0D1HC 46871782 IC50 = 370 nM T13201 D0D2JA 2734377 Ki = 6000 nM T13201 D0D4OV 20043772 Ki = 378 nM T13201 D0D5XC 101753 Ki = 8700 nM T13201 D0D6UR 12394434 Ki = 12400 nM T13201 D0DY9U 23645365 Ki = 74 nM T13201 D0E0RW 69894 Ki = 14000 nM T13201 D0E3VJ 25154731 Ki = 1890 nM T13201 D0E8CC 18794 Ki = 15 nM T13201 D0EH0S 52943164 Ki > 100000 nM T13201 D0EJ9B 66827 Ki = 58.6 nM T13201 D0EX9Q 10881548 Ki = 1500 nM T13201 D0EY2F 52949920 Ki > 100000 nM T13201 D0F3UR 690836 Ki > 50000 nM T13201 D0F7KC 14116752 Ki > 100000 nM T13201 D0F7QZ 5702628 Ki = 12500 nM T13201 D0F7SO 94464 Ki = 21000 nM T13201 D0FD8G 6011033 Ki = 10700 nM T13201 D0FU0K 23354226 Ki > 10000 nM T13201 D0G0BJ 51000408 Ki > 50000 nM T13201 D0G0FJ 11206245 Ki = 24000 nM T13201 D0G0OP 44423685 Ki = 9800 nM T13201 D0G0ZI 403788 Ki = 5690 nM T13201 D0G3BI 25090 Ki = 6800 nM T13201 D0G3TK 5280863 Ki > 10000 nM T13201 D0G6OW 23675285 Ki = 74000 nM T13201 D0G9NE 11659798 Ki = 880 nM T13201 D0GQ9A 44593649 Ki = 31700000 nM T13201 D0H3NS 10752 Ki = 9300 nM T13201 D0HN0R 11623958 Ki = 3560 nM T13201 D0I5YQ 44405178 Ki = 1130 nM T13201 D0I8DW 612414 Ki = 18 nM T13201 D0IB3K 5320686 Ki > 10000 nM T13201 D0IU3X 44405186 Ki = 273 nM T13201 D0J1PZ 2723687 Ki = 4500 nM T13201 D0J2AE 7377 Ki = 25000 nM T13201 D0J3SP 11718391 Ki = 4.1 nM T13201 D0J7GU 46703929 Ki = 9030 nM T13201 D0J7KJ 52940758 Ki > 100000 nM T13201 D0K1FG 5411574 Ki > 100000 nM T13201 D0K3LN 3510137 Ki = 19300 nM T13201 D0K4IH 687887 Ki = 1230 nM T13201 D0K5NQ 10421755 Ki = 8 nM T13201 D0KB6T 721954 Ki = 3300 nM T13201 D0KZ2D 11638641 Ki = 810 nM T13201 D0L1AV 45273021 IC50 = 23000000 nM T13201 D0L2GD 60167587 Ki = 6900 nM T13201 D0L4FM 11030308 Ki = 2.1 nM T13201 D0L5TZ 20195365 Ki = 243000 nM T13201 D0L5XK 92249 Ki = 5560 nM T13201 D0L8ZG 79799 Ki = 278000 nM T13201 D0LC0F 96876 Ki = 215 nM T13201 D0LJ5P 44457221 Ki = 1080 nM T13201 D0LU4S 156219 Ki = 37000 nM T13201 D0M3PO 69561 Ki = 5800 nM T13201 D0M4EV 18975977 Ki = 20 nM T13201 D0M5MI 4306515 IC50 > 100000 nM T13201 D0M6RM 7365 Ki = 31.7 nM T13201 D0M7VN 44392435 Ki = 28000 nM T13201 D0N0JL 1023 Ki = 25800000 nM T13201 D0N1AW 45485270 Ki = 99 nM T13201 D0N5KX 44391625 Ki > 20 nM T13201 D0N7WP 44520903 Ki = 75 nM T13201 D0N8LR 847760 Ki = 19700 nM T13201 D0NN3Q 78105 Ki = 3900 nM T13201 D0NS0E 220188 Ki > 10000 nM T13201 D0O0UE 729977 Ki = 7.6 nM T13201 D0O1QT 93505 Ki = 55 nM T13201 D0O4KL 11640067 Ki = 770 nM T13201 D0O6ZD 14101447 Ki > 100000 nM T13201 D0O8WV 11536481 Ki = 825 nM T13201 D0O9VU 44520901 Ki = 67 nM T13201 D0OC4B 5357479 Ki > 10000 nM T13201 D0OI1H 72894 Ki = 45400 nM T13201 D0OT5L 1631814 Ki = 23100 nM T13201 D0P6AM 3526523 Ki = 186 nM T13201 D0PA5L 44380941 Ki = 34 nM T13201 D0Q0EK 318174 Ki = 2950 nM T13201 D0Q0XO 4258082 Ki = 17650 nM T13201 D0Q1EI 3084733 Ki = 9650 nM T13201 D0Q2XB 75928 Ki = 38810 nM T13201 D0Q5VB 46704078 Ki = 5620 nM T13201 D0Q7DJ 10742 Ki = 4150 nM T13201 D0R4KQ 46704077 Ki = 10300 nM T13201 D0R4WJ 16129778 Ki = 75900 nM T13201 D0R7QY 127676 Ki = 37 nM T13201 D0RB0D 44268050 Ki = 3720 nM T13201 D0RK7J 235259 Ki = 14600 nM T13201 D0S0RK 10680 Ki = 1880 nM T13201 D0S1OY 10946908 Ki = 3700 nM T13201 D0S2II 308405 Ki = 311 nM T13201 D0S3RZ 9954405 Ki = 6 nM T13201 D0S4NO 25154730 Ki = 7010 nM T13201 D0S6CO 17655 IC50 = 430 nM T13201 D0S9YX 5280373 Ki > 10000 nM T13201 D0SF3B 11529486 Ki = 875 nM T13201 D0SY2M 5281708 Ki > 10000 nM T13201 D0T0YI 378 IC50 = 330 nM T13201 D0T2VH 44571846 Ki = 5540 nM T13201 D0T2YZ 3253857 Ki = 23500 nM T13201 D0T3NP 7456 Ki = 2600 nM T13201 D0T6VB 521293 Ki = 700 nM T13201 D0T8SN 12033284 Ki = 14 nM T13201 D0T9BB 52950111 Ki > 100000 nM T13201 D0TY8X 31036 Ki = 95 nM T13201 D0U1AN 521359 Ki = 5000 nM T13201 D0U4BB 10748 Ki = 5900 nM T13201 D0UM1I 12554666 Ki = 7910 nM T13201 D0UN0E 12195854 Ki = 357 nM T13201 D0V0FY 52946831 Ki > 100000 nM T13201 D0V5OW 46907400 Ki = 9510 nM T13201 D0V9EN 689043 Ki = 2380 nM T13201 D0VD7H 84724 IC50 = 2600 nM T13201 D0W1AW 4234241 Ki = 63.4 nM T13201 D0W1OR 7424 Ki = 550 nM T13201 D0W9VC 670143 Ki = 61 nM T13201 D0X0PO 20043771 Ki = 136 nM T13201 D0X0RE 6019835 Ki = 12100 nM T13201 D0X1MY 2723847 Ki = 7100 nM T13201 D0X5HL 15107 Ki > 500000 nM T13201 D0X6IE 4422372 Ki = 100 nM T13201 D0X9LJ 788811 Ki = 870 nM T13201 D0XK7G 10445302 Ki = 30 nM T13201 D0XL5K 67944 Ki = 95 nM T13201 D0Y1XM 44423686 Ki = 520000 nM T13201 D0Y3TZ 370 Ki = 3200 nM T13201 D0Y7HG 5281616 Ki > 10000 nM T13201 D0YD9F 822774 Ki = 103 nM T13201 D0YU8J 1502014 Ki = 9800 nM T13201 D0YZ5G 5281416 Ki > 10000 nM T13201 D0Z1CL 79599 Ki = 11700 nM T13201 D0Z1HY 67136 Ki = 8400 nM T13201 D0Z5GE 44520902 Ki = 263 nM T13201 D0Z6TM 3558590 Ki = 3900 nM T13201 D0ZC3W 6269 Ki = 78500 nM T90989 D04LVK 57379345 IC50 = 950 nM T90989 D0H0EQ 24826799 IC50 = 7.1 nM T90989 D03LWG 53235510 IC50 = 0.82 nM T90989 D07EHV 44814409 IC50 > 10000 nM T90989 D07HPJ 11476171 IC50 = 5000 nM T90989 D08EQD 118036971 IC50 = 1.9 nM T90989 D0D4VV 46944259 IC50 = 3.2 nM T90989 D0D6XT 118029202 IC50 < 1.2 nM T90989 D0E3TC 44259 IC50 = 107 nM T90989 D0H9FR 118295624 IC50 = 19.3 nM T90989 D0NW0T 67462786 IC50 = 5.7 nM T90989 D0XT0W 66555680 IC50 = 290 nM T90989 D03BNU 59604787 IC50 > 10000 nM T90989 D08DBE 10344820 Ki = 217 nM T90989 D0T3ME 156422 IC50 = 7000 nM T90989 CPT61U 5328112 IC50 = 560 nM T90989 CFHA86 9797013 IC50 > 10000 nM T90989 CACS26 11561968 Ki > 2000 nM T90989 CU0E8O 11690457 Ki > 2000 nM T90989 CP7AH3 11755812 IC50 = 50000 nM T90989 C2B5XF 49765254 IC50 > 10000 nM T90989 CJZ5A0 49840306 IC50 > 10000 nM T90989 C90ANW 50939489 IC50 = 340 nM T90989 CEQN27 52936621 Ki > 1000 nM T90989 C09SDH 53257410 IC50 > 10000 nM T90989 C4F6SR 53348188 IC50 = 189 nM T90989 C8NA4L 53384644 IC50 > 30000 nM T90989 CUPT85 54406017 IC50 > 10000 nM T90989 C8P6RD 57505528 IC50 > 10000 nM T90989 CPU2E3 59737752 IC50 = 29 nM T90989 C1MR8Q 60097495 IC50 > 1000 nM T90989 C9O4GF 66555232 IC50 = 250 nM T90989 CL3EN2 66556938 IC50 = 490 nM T90989 C1HSE0 67035086 IC50 = 2800 nM T90989 CWI6K5 67035106 IC50 > 10000 nM T90989 C38RGB 67035556 IC50 > 10000 nM T90989 CV63UL 67240318 IC50 > 10000 nM T90989 CO6W9D 68004741 IC50 = 13 nM T90989 CB6U7F 68005465 IC50 = 26 nM T90989 CK83VI 68005486 IC50 = 720 nM T90989 C1RJ7Y 68005600 IC50 = 240 nM T90989 COX3U9 68005621 IC50 = 130 nM T90989 CEXN58 68005732 IC50 = 220 nM T90989 C8I7GC 68293638 IC50 > 10000 nM T90989 CD56XK 68293660 IC50 > 10000 nM T90989 C9OQ2I 72710839 IC50 = 3 nM T90989 CQ5E3H 73707531 IC50 = 22 nM T90989 CRQO23 86293280 IC50 = 2772 nM T90989 C4OC7T 86293469 IC50 = 526 nM T90989 CPG3A5 86302574 IC50 > 30000 nM T90989 CF27DP 91825767 IC50 = 32 nM T90989 COR1E4 118036202 IC50 = 6.3 nM T90989 C6ZT7E 118036250 IC50 = 13 nM T90989 CMVJ36 118036287 IC50 = 175 nM T90989 CGXP67 118036351 IC50 = 916 nM T90989 C7P8NT 118036414 IC50 = 11 nM T90989 CO4UR1 118036466 IC50 = 45 nM T90989 CR9S7W 118036565 IC50 = 4.5 nM T90989 CND4C7 118036674 IC50 = 660 nM T90989 C84BWP 118036727 IC50 = 42 nM T90989 C4TH7L 118036769 IC50 = 27 nM T90989 C7ZE6W 118036804 IC50 = 1.2 nM T90989 C24JLP 118036824 IC50 = 1.3 nM T90989 CUTW04 118036840 IC50 = 1.6 nM T90989 CA6DN5 118036877 IC50 = 0.7 nM T90989 CUQX28 118036931 IC50 = 16 nM T90989 CZCO25 118036941 IC50 = 140 nM T90989 CIK29M 118036948 IC50 = 1.1 nM T90989 C8BL6F 118036962 IC50 = 17 nM T90989 C1G6DN 118037014 IC50 = 300 nM T90989 COQ2G9 118037084 IC50 = 33 nM T90989 CVB8Q7 118728412 IC50 = 20 nM T90989 CH1B5J 118893306 IC50 = 52.7 nM T90989 C08KEM 122179540 IC50 = 5900 nM T90989 C3AJ4C 122179546 IC50 = 9200 nM T90989 CG0RP7 122179547 IC50 = 5300 nM T90989 C1A0SQ 122179548 IC50 = 4400 nM T90989 CSL75U 122573595 IC50 = 6.5 nM T90989 CIG5F7 122573596 IC50 = 7.4 nM T90989 CLM7K3 122604539 IC50 = 13 nM T90989 C01JHI 122604566 IC50 = 3 nM T90989 C1E4AR 122604567 IC50 = 4 nM T90989 CQJZ70 122604640 IC50 = 4 nM T90989 CMQ9V3 122606542 IC50 = 8 nM T90989 CY30FL 123752658 IC50 = 5.5 nM T90989 C9SI5T 127047969 IC50 = 52.7 nM T90989 C2LWZ1 129318964 IC50 > 10000 nM T90989 C9Y5TL 132156608 IC50 = 9.5 nM T90989 CUO0C5 132156633 IC50 = 1.5 nM T90989 CUW5L2 132156656 IC50 = 11.1 nM T90989 CT3DM9 132156669 IC50 = 3.5 nM T90989 CY35PA 132156727 IC50 = 2.1 nM T90989 C0R2MF 132156728 IC50 = 1.4 nM T90989 CZN5W1 132156731 IC50 = 71 nM T90989 CQB04N 132156743 IC50 = 4.7 nM T90989 C53HPM 132156749 IC50 = 7.5 nM T90989 C3UA1J 132156758 IC50 = 1 nM T90989 CJ7B4Q 132156777 IC50 = 38 nM T90989 C8A7XK 132156780 IC50 = 5.3 nM T90989 CBWE03 132156803 IC50 = 4.6 nM T90989 CO3P6X 132156815 IC50 = 2.7 nM T90989 C95HIB 132156818 IC50 = 1.3 nM T90989 C3CD6R 132156853 IC50 = 4.6 nM T90989 C3V5TF 132245876 IC50 > 100 nM T90989 CXA84S 132245879 IC50 = 3.8 nM T90989 C8HPV6 132245890 IC50 = 6.2 nM T90989 C4F9YW 132245892 IC50 = 5.4 nM T90989 C5QZ7A 132245893 IC50 = 55.4 nM T90989 CA3IV9 132245894 IC50 = 38.8 nM T90989 C95XEY 132245912 IC50 = 327.3 nM T90989 CIJ6Y0 132245918 IC50 = 64.3 nM T90989 CKW5S9 132245920 IC50 = 489 nM T90989 CX3ZV1 132245921 IC50 = 33.2 nM T90989 C8U1MG 132245924 IC50 = 145.7 nM T90989 C6H3JS 132245929 IC50 = 35.6 nM T90989 CPN39H 132245933 IC50 = 25.9 nM T90989 C8U0OD 132245935 IC50 = 19.4 nM T90989 C7VW5M 132245939 IC50 = 1.7 nM T90989 CMER63 132245964 IC50 = 179.5 nM T90989 CRIN01 132245965 IC50 = 31.2 nM T90989 C5XLN0 132245967 IC50 = 90.6 nM T90989 CFY9W5 132245971 IC50 = 312.9 nM T90989 CULE97 132245973 IC50 = 155 nM T90989 C5K7YE 132246005 IC50 > 1000 nM T90989 CR85IS 132246032 IC50 = 145 nM T90989 C2JPX7 132246037 IC50 = 42.8 nM T90989 C4YSB5 132246051 IC50 = 19.4 nM T90989 CK9W4F 134135741 IC50 = 4100 nM T90989 CMA60G 134144799 IC50 > 50000 nM T90989 C3MN6B 134144868 IC50 = 3100 nM T90989 CEZH84 134146580 IC50 = 110 nM T90989 C1DF4R 134147544 IC50 = 740 nM T90989 C95NCV 134151662 IC50 = 200 nM T90989 CX7YE1 134155961 IC50 = 85 nM T90989 CE38MW 134156584 IC50 = 160 nM T90989 CVI25K 134157526 IC50 = 730 nM T90989 C71CBJ 134255819 IC50 = 1.7 nM T90989 CBGO29 134255820 IC50 = 1.2 nM T90989 CI8L9W 134255882 IC50 = 5 nM T90989 C5UBG7 134255896 IC50 = 1 nM T90989 CVE4X3 134457519 IC50 = 188 nM T90989 CO1IL0 134457555 IC50 = 3.8 nM T90989 CB15KN 134457556 IC50 = 24.9 nM T90989 CCFS35 134457606 IC50 = 4.8 nM T90989 CEAH09 134457612 IC50 = 8.5 nM T90989 C1P9KY 134457618 IC50 = 2.6 nM T90989 CGAV72 134457621 IC50 = 5.3 nM T90989 CJYX87 134457890 IC50 > 10000 nM T90989 CWZ1L4 135316948 IC50 = 383 nM T90989 C5B6XD 135316952 IC50 = 166 nM T90989 CWEP52 135316962 IC50 = 186 nM T90989 CW5KL0 135316982 IC50 = 296 nM T90989 C6E5FP 135317017 IC50 = 269 nM T90989 CCTW97 135317286 IC50 = 68.7 nM T90989 CH2JK6 135317468 IC50 = 47.8 nM T90989 CFE0X7 135317546 IC50 = 452 nM T90989 C0JM1W 135317567 IC50 = 44.2 nM T90989 CI2L5A 135317791 IC50 = 78.1 nM T90989 CJZ59L 135317844 IC50 = 180 nM T90989 C45XNW 135318783 IC50 = 79.2 nM T90989 CS63IO 135476717 IC50 = 610 nM T90989 C4WX3I 135486449 IC50 > 20000 nM T90989 CTJ48K 135524085 IC50 = 6800 nM T90989 CUT1W7 135524168 IC50 > 10000 nM T90989 CYXU86 136180312 IC50 > 20000 nM T90989 C9MHA4 136180313 IC50 > 20000 nM T90989 CDT7E4 136211077 IC50 = 6.1 nM T90989 C7PNC4 136243300 IC50 > 20000 nM T90989 CUN1I4 136243344 IC50 > 20000 nM T90989 C68IKN 136243473 IC50 > 20000 nM T90989 CH4T8M 136961363 IC50 > 20000 nM T90989 C7N8EG 136961364 IC50 > 20000 nM T90989 CRPQ98 136961365 IC50 > 20000 nM T90989 CSZ16N 136961366 IC50 > 20000 nM T90989 CB9D7F 136961367 IC50 > 20000 nM T90989 CEPT42 136961368 IC50 > 20000 nM T90989 C25ERN 137631967 IC50 = 7.4 nM T90989 C0J6IC 137633737 IC50 > 1000 nM T90989 CNX0F9 137634126 IC50 = 166.9 nM T90989 C2K8LT 137636345 IC50 = 38.7 nM T90989 CF7O2C 137636828 IC50 = 43.4 nM T90989 CPR60M 137637024 IC50 = 25.6 nM T90989 C06JRX 137637094 IC50 = 299.4 nM T90989 C6BIO8 137637138 IC50 = 3500 nM T90989 CMCI72 137638094 IC50 = 152.4 nM T90989 C3OVJ8 137638489 IC50 = 27 nM T90989 C7J8FB 137639540 IC50 = 669.2 nM T90989 CFUX56 137640843 IC50 = 148 nM T90989 C5E6NQ 137643062 IC50 = 465.7 nM T90989 CY8L5M 137644036 IC50 = 3 nM T90989 C0CTB5 137644554 IC50 = 72.9 nM T90989 CS3TU7 137644762 IC50 = 24 nM T90989 C79SUZ 137646264 IC50 = 8.2 nM T90989 C7P5AX 137646321 IC50 = 202.3 nM T90989 CSJ4N3 137646379 IC50 = 1200 nM T90989 C7CA9N 137646692 IC50 = 12.3 nM T90989 CGF7X2 137647982 IC50 > 1000 nM T90989 C7EZP8 137649394 IC50 > 10000 nM T90989 CHSB74 137650627 IC50 = 273.5 nM T90989 C1DK0P 137651391 IC50 = 93.3 nM T90989 C0MZ1W 137652333 IC50 = 7.5 nM T90989 CBAF08 137653174 IC50 > 10000 nM T90989 CV5H3Z 137657932 IC50 = 61.7 nM T90989 C7SEK1 137658232 IC50 = 17.1 nM T90989 CQF74K 137658987 IC50 = 22.7 nM T90989 C8DZ6L 137659285 IC50 = 28.1 nM T90989 C9UMG4 137660300 IC50 > 1000 nM T90989 CTJV46 137660921 IC50 = 6 nM T90989 CW9U3A 137661140 IC50 = 98 nM T90989 CM3UF7 137700779 IC50 > 10000 nM T90989 CSRI06 138547901 IC50 = 23.1 nM T90989 C04KQV 138617497 IC50 = 82.7 nM T90989 CUXO19 138617501 IC50 = 5.3 nM T90989 CZ2XH5 139187793 IC50 = 43 nM T90989 CUH2G6 139554482 IC50 = 1.5 nM T90989 CO9P7G 145351804 IC50 > 1000 nM T90989 C29XUO 145945978 IC50 > 200 nM T90989 CB3Z1W 145949428 IC50 = 1076 nM T90989 C5VSC7 145956704 IC50 = 866 nM T90989 C8ENC3 145979734 IC50 > 10000 nM T90989 CIA9B7 145980214 IC50 = 23 nM T90989 C93AOR 145980752 IC50 = 2.2 nM T90989 CX7ZE5 145981170 IC50 = 5200 nM T90989 CEH13K 145981554 IC50 = 790 nM T90989 CTE48L 145985844 IC50 > 10000 nM T90989 CSM23R 145988105 IC50 = 9500 nM T90989 C8ED6I 145988852 IC50 > 10000 nM T90989 C10FNU 145990947 IC50 = 4400 nM T90989 CS6KH7 145992430 IC50 > 10000 nM T90989 CJMQ90 145993820 IC50 = 3.2 nM T90989 CS7TD1 145993995 IC50 = 21 nM T90989 CN7EF3 145996526 IC50 > 1000 nM T90989 C9X8LP 155513025 IC50 = 85.2 nM T90989 C2MD1Q 155513187 IC50 > 10000 nM T90989 CL75PC 155515231 IC50 = 9.1 nM T90989 C86HPW 155518524 IC50 = 11000 nM T90989 C2HL6O 155519199 IC50 = 9.4 nM T90989 CX37HC 155537699 IC50 > 1000 nM T90989 C0BRU3 155547256 IC50 = 1.3 nM T90989 C9WN5D 155554550 IC50 = 78.9 nM T90989 C21DWP 155564268 IC50 = 94.3 nM T90989 CIN82D 155568305 IC50 = 779 nM T90989 D02BXJ 46864270 IC50 = 34 nM T90989 D06HVH 54613583 IC50 > 10000 nM T90989 D0L0SP 6579 IC50 = 938 nM T90989 D0R2WK 16038120 IC50 = 16 nM T82668 D07JBL 67962992 Ki = 23 nM T82668 D09JPJ 71717745 Ki = 41 nM T82668 D0RR5C 67963001 IC50 = 329 nM T82668 D0SZ7H 67813781 Ki = 1.9 nM T82668 C4U2LE 11147888 IC50 > 10000 nM T82668 CI0R3X 12643457 IC50 > 10000 nM T82668 C4DZ1K 21787167 IC50 = 3280 nM T82668 C2UP5H 22868923 Ki = 14 nM T82668 CBIC15 22868926 IC50 > 10000 nM T82668 C2E6PT 22868930 IC50 = 29 nM T82668 CAPS68 46829291 IC50 = 910 nM T82668 C40LGZ 49864178 IC50 = 1500 nM T82668 CFKA48 53253721 IC50 = 29 nM T82668 CVDK24 53253769 IC50 = 174 nM T82668 C8OEX2 53254439 IC50 = 319 nM T82668 C8D3IV 53254440 IC50 = 45 nM T82668 CHU60C 53254441 IC50 = 30 nM T82668 CW4P5Y 53254442 IC50 = 36 nM T82668 CAJ1G9 53254526 Ki = 7.7 nM T82668 CF76GZ 53254527 IC50 = 37 nM T82668 C8UBW9 53254677 IC50 = 572 nM T82668 C1EO6K 53254679 IC50 = 1050 nM T82668 CQKC01 53254681 IC50 = 252 nM T82668 C95KSM 59627033 Ki = 1.6 nM T82668 C0V8PC 59627051 IC50 = 40 nM T82668 CM8BC1 59627101 Ki = 7.1 nM T82668 C5DL2Y 59627133 IC50 = 179 nM T82668 C6YPN0 59627156 IC50 = 349 nM T82668 CA8G7O 59627182 IC50 = 219 nM T82668 CLN87P 62707349 IC50 > 10000 nM T82668 CV6XI8 67962969 Ki = 22 nM T82668 C8U7CM 67963007 Ki = 12 nM T82668 CV5R6U 71059324 Ki = 32 nM T82668 CQPD97 71059651 Ki = 48 nM T82668 CJG3N6 71717990 Ki = 1.66 nM T82668 CW2RE4 72714743 Ki = 5.1 nM T82668 CDGT12 72714838 Ki = 81.5 nM T82668 CY53GN 72714928 IC50 = 84 nM T82668 C59RAW 90667360 Ki = 16.7 nM T01865 CC3FJ6 9996876 Ki = 26000 nM T01865 CLQ5I2 13365345 Ki = 19000 nM T01865 C95WBH 13365350 Ki = 23000 nM T01865 CZN37R 13365355 Ki = 30000 nM T01865 C8KJ3G 13365369 Ki > 500000 nM T01865 CEJ51X 44408132 Ki > 500000 nM T01865 CEQ32O 44408134 Ki > 500000 nM T01865 CJ38RE 44408135 Ki = 130000 nM T01865 CO9TW6 44408159 Ki > 500000 nM T01865 CWE1O8 44408160 Ki > 500000 nM T01865 CA3P5J 44408175 Ki = 140000 nM T01865 C5OE7L 44408183 Ki = 36000 nM T01865 C1AT5Z 44408187 Ki = 37000 nM T01865 CA19UM 44408261 Ki = 64000 nM T01865 C2DC6S 44408262 Ki = 148000 nM T01865 C9NZO7 44408268 Ki > 500000 nM T01865 CPLK96 44408297 Ki = 41000 nM T01865 C23ZXG 44408299 Ki = 49000 nM T01865 CS7LG3 44408300 Ki = 81000 nM T01865 C0O6PG 44408301 Ki > 500000 nM T01865 CU5VW1 44408303 Ki = 590000 nM T01865 C5VD9J 44408385 Ki < 500000 nM T01865 CI1C0Q 44408489 Ki = 30000 nM T01865 C3M9FL 44408498 Ki = 32000 nM T01865 CAFS82 44408566 Ki = 540000 nM T01865 C0A8XY 44442293 Ki > 500000 nM T01865 CX3J1L 44442294 Ki > 500000 nM T01865 CFX9N2 44442295 Ki > 500000 nM T01865 C4NG1C 44442296 Ki > 500000 nM T01865 C5B2GA 44442297 Ki = 2000 nM T01865 C0THJ5 44442298 Ki = 1500000 nM T01865 CAH90M 44442299 Ki = 2000000 nM T48330 D01CRB 6057 IC50 = 68000 nM T48330 D05EJG 6305 IC50 = 160000 nM T48330 D08HVR 6047 IC50 = 100000 nM T48330 D0R1CR 6140 IC50 = 69000 nM T48330 D0N0KW 84815 IC50 = 120000 nM T48330 CWFP01 71098 IC50 = 380000 nM T48330 C5X2WA 71563 IC50 > 50000000 nM T48330 CJ1C7V 92105 IC50 = 190000 nM T48330 CJ0RF7 94206 IC50 > 3000000 nM T48330 C4RGU9 152953 IC50 = 69000 nM T48330 CD41MN 193138 IC50 = 170000 nM T48330 C7JDZ1 439524 IC50 = 220000 nM T48330 C6PG0C 736026 IC50 = 260000 nM T48330 CNXW98 2724754 IC50 = 130000 nM T48330 CTM90S 2761499 IC50 = 160000 nM T48330 CDW5A8 2762277 IC50 = 470000 nM T48330 C9CP4S 7009701 IC50 = 100000 nM T48330 C6FYC2 7023409 IC50 = 810000 nM T48330 CT4X6Y 10060246 IC50 = 6600 nM T48330 C1BE9O 11521308 IC50 = 92000 nM T48330 CQEZ46 12042114 IC50 = 340000 nM T48330 CRG8J4 12085165 IC50 = 240000 nM T48330 C2K7JL 18656092 IC50 = 36000 nM T48330 CS5VJ8 22854522 IC50 = 130000 nM T48330 C7A4UI 24853505 IC50 = 790 nM T48330 C3CX6Y 45116514 IC50 = 260000 nM T48330 CH97TV 53754520 IC50 = 101000 nM T48330 CR7M3V 53819050 IC50 = 9100 nM T48330 CH3O5F 57039748 IC50 = 7300 nM T48330 CN1B5D 57155616 IC50 = 17000 nM T48330 C7K1TA 66743594 IC50 = 160000 nM T48330 CML86J 67059715 IC50 = 83000 nM T48330 C6RF5A 68530773 IC50 = 110000 nM T48330 CMB9N1 94905321 IC50 > 1000000 nM T48330 CX6C2O 145983064 IC50 = 29000 nM T48330 C1L6WX 145983243 IC50 = 27700 nM T48330 C8UD2J 145983285 IC50 = 32380 nM T48330 C67FNE 145983610 IC50 = 680000 nM T48330 CH5G1A 145984011 IC50 = 76000 nM T48330 CDI23V 145984714 IC50 = 95000 nM T48330 C15EMU 145985040 IC50 = 150000 nM T48330 CWG62S 145985227 IC50 = 96000 nM T48330 CD1MX7 154730690 IC50 = 18200 nM T48330 CZG8T2 155519448 IC50 > 1000000 nM T48330 C7W9YE 155544142 IC50 = 980 nM T48330 CT9W2I 155552110 IC50 > 1000000 nM T48330 CIX4G6 155566772 IC50 = 440000 nM T48330 D00XUE 712421 IC50 = 200000 nM T48330 D05BOD 115288 IC50 = 112000 nM T48330 D05XGI 6950578 IC50 = 130000 nM T48330 D08CBB 9060 IC50 = 380000 nM T48330 D0B3LN 71567 IC50 = 46000 nM T48330 D0I8SK 6306 IC50 = 140000 nM T48330 D0LL5V 6287 IC50 = 68000 nM T48330 D0PG8L 71083 IC50 = 460000 nM T48330 D0PO8E 6137 IC50 = 170000 nM T48330 D0T6UL 6274 IC50 = 110000 nM T48330 D0W4MZ 6106 IC50 = 85000 nM T31992 D00STL 644241 Ki = 223 nM T31992 D01MUR 68844 Ki = 24 nM T31992 D03RTS 2662 Ki = 689 nM T31992 D03UOT 785 Ki = 42000 nM T31992 D05OFX 219078 Ki = 473 nM T31992 D05UYW 5284549 Ki = 27 nM T31992 D07HBX 338 Ki = 49800 nM T31992 D07INV 3295 Ki = 2.5 nM T31992 D07VDZ 5284627 Ki = 1460 nM T31992 D09NIA 2732 Ki = 4130 nM T31992 D09VAZ 5565 Ki = 12100 nM T31992 D0AZ3C 5291 Ki = 468 nM T31992 D0AZ8C 5213 Ki = 11640 nM T31992 D0C2II 4100 Ki = 43 nM T31992 D0C8FX 3005837 Ki = 2910 nM T31992 D0E1SW 1986 Ki = 5.7 nM T31992 D0H8FH 3702 Ki = 4950 nM T31992 D0J4GO 3038 Ki = 345 nM T31992 D0J7RK 36811 Ki = 12020 nM T31992 D0K0OZ 5702160 Ki = 677.2 nM T31992 D0K1QD 3998 Ki = 3200 nM T31992 D0K8KX 5280343 Ki = 5410 nM T31992 D0L4JT 5333 Ki = 5400 nM T31992 D0L6DA 119607 Ki = 107 nM T31992 D0OT0O 44561 Ki = 3600000 nM T31992 D0PQ3G 3440 Ki = 52 nM T31992 D0SH3I 387447 Ki = 3280 nM T31992 D0U5QK 1983 Ki = 10600 nM T31992 D0VM2L 68740 IC50 = 92 nM T31992 D0Y2IZ 5560 Ki = 3450 nM T31992 D0Z3EI 6038 Ki = 36 nM T31992 D04IIU 216468 Ki = 104 nM T31992 D05NJI 5287541 Ki = 755 nM T31992 D08BXT 1102 Ki = 1000 nM T31992 D0L6HN 996 Ki = 11500 nM T31992 D0U3EP 445154 Ki = 830 nM T31992 D0V0UK 82267 Ki = 750000 nM T31992 D03SLR 445858 Ki = 9430 nM T31992 D0NH9P 135 Ki = 6160 nM T31992 D0LD9S 1103 Ki = 860 nM T31992 CI0WH9 72 Ki = 690 nM T31992 CU12QE 1203 Ki = 11550 nM T31992 C6O0MZ 1491 Ki = 70000 nM T31992 C5L7VX 2871 Ki = 4140 nM T31992 CQ0D8J 3469 Ki = 67000 nM T31992 CJ2F6P 5056 Ki = 1950 nM T31992 CDJ4K6 5987 Ki = 1090000 nM T31992 CUP2F4 7043 Ki = 6830 nM T31992 C1CVT7 7121 Ki = 740 nM T31992 C6NC4O 7414 Ki = 4550 nM T31992 C6QYD8 8434 Ki = 7700 nM T31992 CHP7I1 9016 Ki = 6790 nM T31992 CLYZ50 9338 Ki = 6500 nM T31992 CV5PC3 11568 Ki = 7200 nM T31992 CNI85U 15109 Ki = 550 nM T31992 CQ4C5U 16523 Ki = 860 nM T31992 CNGB21 20098 Ki = 830 nM T31992 C3LA1Z 20161 Ki = 820 nM T31992 C4OU6D 35703 Ki = 8900 nM T31992 CY2GU3 60582 Ki = 6.1 nM T31992 C0ZK7U 67284 Ki = 630 nM T31992 CVI38F 69809 Ki = 9790 nM T31992 CTMF08 75076 Ki = 780 nM T31992 C0I4UT 75077 Ki = 800 nM T31992 CE5RZ1 76509 Ki = 740 nM T31992 C9V0ME 77547 Ki = 860 nM T31992 C6TS8J 77548 Ki = 770 nM T31992 CX47BZ 78479 Ki = 36000 nM T31992 C5BFK4 87432 Ki = 820 nM T31992 CN19UT 129695 Ki = 1030 nM T31992 CCK5Y6 133125 Ki = 4 nM T31992 CVB67D 134560 Ki = 13 nM T31992 CSMP84 219987 Ki = 48800 nM T31992 C3QV5H 287064 Ki = 890 nM T31992 CT3ZU4 388776 Ki = 6700 nM T31992 CH21KA 389641 Ki = 85000 nM T31992 C6CQO3 389642 Ki = 115000 nM T31992 CNPZ40 394897 Ki = 7.5 nM T31992 CC54LQ 450256 IC50 > 10000 nM T31992 C49CNT 519869 Ki = 760 nM T31992 CYGK68 676946 Ki = 800 nM T31992 CF93TC 821388 Ki = 740 nM T31992 C8SN5L 889524 Ki = 684 nM T31992 CEN67I 897592 Ki = 643 nM T31992 C9DY2L 1488548 Ki = 35500 nM T31992 CE2GR3 2900806 Ki = 34000 nM T31992 CME74N 2904589 Ki = 644 nM T31992 C4E5VQ 4447263 Ki = 65 nM T31992 C96LCZ 4476238 Ki = 78 nM T31992 CLSY09 4626049 Ki = 820 nM T31992 C3GDR0 4634582 Ki = 71 nM T31992 CCB9Z5 4656684 Ki = 82 nM T31992 CX8C3P 4961927 Ki = 3.7 nM T31992 C4OAL9 5070078 Ki = 6400 nM T31992 CI8JY0 5172475 Ki = 245 nM T31992 CY9IV8 5223338 Ki = 5.5 nM T31992 CZS0G5 5276565 IC50 = 7461 nM T31992 C3JN0F 5277465 IC50 = 8214 nM T31992 CRJK67 5277481 IC50 = 911 nM T31992 CYF7S5 5277490 IC50 > 10000 nM T31992 CI58XK 5319562 Ki = 830 nM T31992 C9L8AX 6537802 Ki = 16 nM T31992 C65FRB 6852128 Ki = 4.1 nM T31992 CKCM96 7463376 Ki = 3280 nM T31992 CDCP43 7766335 Ki = 780 nM T31992 CY47OI 9998322 Ki = 76 nM T31992 CF6RN0 10018880 Ki = 34.3 nM T31992 C69DPZ 10068042 IC50 = 3310 nM T31992 CD58EL 10083644 Ki = 810 nM T31992 C3HBY6 10375558 Ki = 3255 nM T31992 C73KXU 10586607 Ki = 41 nM T31992 C9TSQ6 10632698 Ki = 3800 nM T31992 C6D2TJ 10712038 Ki = 25 nM T31992 C8C6ER 11069133 Ki = 0.9 nM T31992 CHC42Y 11245700 Ki = 13 nM T31992 CHA0V5 11321514 Ki = 770 nM T31992 C8PM3Z 11353795 Ki = 33 nM T31992 CFER43 11467281 Ki = 41 nM T31992 CV7HN1 11795548 Ki = 13 nM T31992 C45NRP 11851425 Ki = 94 nM T31992 CZD0B3 11974341 Ki = 11 nM T31992 CC8AI5 11974342 Ki = 71 nM T31992 C27HSO 11974343 Ki = 76 nM T31992 CCM17V 11974451 Ki = 55 nM T31992 CX4IJ0 11974452 Ki = 103 nM T31992 C59UEI 11974453 Ki = 64 nM T31992 CYS7X0 11974454 Ki = 78 nM T31992 C09JGZ 11974455 Ki = 64 nM T31992 CS9VL2 11974456 Ki = 71 nM T31992 CP39YI 11974558 Ki = 155 nM T31992 CB97SM 11974559 Ki = 74 nM T31992 CE8WN6 11974560 Ki = 95 nM T31992 C06CBY 11974561 Ki = 75 nM T31992 CU6K0N 11974562 Ki = 10.8 nM T31992 CI7OE1 11974563 Ki = 87 nM T31992 C6Z5DX 11974630 Ki = 78 nM T31992 CW4X9G 11974631 Ki = 134 nM T31992 CEBO65 11974632 Ki = 123 nM T31992 C7TH2X 11974633 Ki = 67 nM T31992 CGQ6B7 11974724 Ki = 73 nM T31992 CHO9T1 11974725 Ki = 10 nM T31992 CB2DY9 11974726 Ki = 101 nM T31992 CC8TS1 11974727 Ki = 105 nM T31992 CDL18J 11974728 Ki = 58 nM T31992 CBC14R 11974729 Ki = 10.9 nM T31992 C7G3YS 11974830 Ki = 10.8 nM T31992 C1C4JW 11974831 Ki = 10.6 nM T31992 CNHD71 12051191 Ki = 7970 nM T31992 CMPA32 12066940 Ki > 500000 nM T31992 CB15KR 12066941 Ki > 500000 nM T31992 C2XBZ3 12070806 Ki = 31 nM T31992 C60EFT 12354987 Ki = 840 nM T31992 CK90BP 12765315 Ki = 9940 nM T31992 CO8WC5 12938307 Ki = 0.93 nM T31992 C8VM1A 13201770 Ki = 700 nM T31992 CQTX49 13738810 IC50 > 10000 nM T31992 CLS53V 14151811 IC50 = 6590 nM T31992 CQ3D9C 14151815 IC50 = 541 nM T31992 CHOG93 14611919 Ki = 48 nM T31992 C76ASY 14787919 Ki > 200000 nM T31992 CH5YR2 15014351 Ki = 5380 nM T31992 C8PMQ9 15729847 Ki > 200000 nM T31992 C8PER5 15938557 Ki > 500000 nM T31992 CC0Z4V 16119626 Ki = 370 nM T31992 CDWU20 17537594 Ki = 7.6 nM T31992 CK7D2I 17748220 Ki = 540 nM T31992 CLY1N4 17757567 Ki = 40400 nM T31992 CQE5K4 18710120 Ki = 7660 nM T31992 CIEH93 19382975 IC50 = 319 nM T31992 C62PKT 19838794 Ki = 42.8 nM T31992 CDU40W 20184392 Ki = 7100 nM T31992 C61KUX 21726402 Ki = 379 nM T31992 CJ4O2E 21806575 Ki = 4.3 nM T31992 C9U4TE 22313850 Ki = 5320 nM T31992 C7V6YP 23665706 Ki = 6.6 nM T31992 C01LHS 24640776 Ki = 37.9 nM T31992 CT8O2Z 24643222 Ki = 41.5 nM T31992 C8BL9O 24762836 Ki = 9340 nM T31992 CK0D4U 24823300 Ki = 50.3 nM T31992 C5W7AC 24823303 Ki = 104 nM T31992 CZMT56 24823304 Ki = 15.8 nM T31992 CUT3V8 24823479 Ki = 20.1 nM T31992 CNR3U7 24866945 IC50 = 7837 nM T31992 CISH83 25186263 Ki = 1030 nM T31992 CU14KG 25258358 Ki = 8530 nM T31992 CQ1WE2 25258360 Ki = 8400 nM T31992 CL5EZ6 25258361 Ki = 8090 nM T31992 COU19V 25258363 Ki = 8370 nM T31992 CRP6F5 25335375 Ki = 19.4 nM T31992 C5EC2T 26535209 Ki = 34.6 nM T31992 CA9UZ7 26773685 Ki = 13.7 nM T31992 CI0K1J 36865965 Ki = 23.8 nM T31992 C6WU8M 42609905 Ki = 5.6 nM T31992 CYJ0H4 43089860 Ki = 41.7 nM T31992 CXJY80 43235186 Ki = 31.4 nM T31992 C82MRL 44144383 Ki = 424 nM T31992 C9J2ME 44395133 Ki = 15.4 nM T31992 CI3O9B 44395149 Ki = 3407 nM T31992 CPB8W7 44395163 Ki = 24.1 nM T31992 CMSJ40 44395790 Ki = 0.47 nM T31992 C5GJ3N 44399351 Ki = 23.5 nM T31992 CZ4DF9 44399462 Ki = 10.4 nM T31992 CU7BK9 44399535 Ki = 17.9 nM T31992 CD5MJ6 44399571 Ki = 9.3 nM T31992 C2T7MB 44399654 Ki = 7.1 nM T31992 CA90GQ 44424362 Ki = 8790 nM T31992 C5HB4P 44424363 Ki > 200000 nM T31992 CK8S7Y 44424364 Ki > 200000 nM T31992 C28QYE 44424366 Ki = 52600 nM T31992 CM3J0U 44430517 Ki = 2350 nM T31992 C9LT7Y 44430518 Ki = 1320 nM T31992 C1VTB6 44430520 Ki = 3500 nM T31992 C2L5MB 44430521 Ki = 630 nM T31992 CVEO17 44430523 Ki = 800 nM T31992 C8MFL1 44430524 Ki = 21 nM T31992 C64APD 44574189 Ki = 3860 nM T31992 CV5XS1 44574190 Ki = 7020 nM T31992 CE0ZS5 44574217 Ki = 8980 nM T31992 C3OYU7 44574218 Ki = 3040 nM T31992 CHJV65 44574219 Ki = 6930 nM T31992 C4FI0H 44574220 Ki = 7050 nM T31992 CM9E2T 44574221 Ki = 5350 nM T31992 C5MCT7 44574248 Ki = 210 nM T31992 CZB19D 44574249 Ki = 6670 nM T31992 C48VUR 44574250 Ki = 3070 nM T31992 CXD9V3 44590306 Ki = 5920 nM T31992 COX6D8 45028566 Ki = 86.1 nM T31992 C80CDA 45028892 Ki = 98.5 nM T31992 C6YHW4 45028893 Ki = 93.8 nM T31992 C23MVW 45269009 IC50 = 780 nM T31992 C0RG8K 45269749 Ki = 7100 nM T31992 CV5RQ3 45484187 Ki = 6700 nM T31992 CTG20B 45485271 Ki = 40 nM T31992 CK4U0V 45485283 Ki = 42 nM T31992 C6ION5 46236927 Ki = 771 nM T31992 C7SFG3 46236928 Ki = 660 nM T31992 CC82QE 46237039 Ki = 7.3 nM T31992 CBCK34 46237040 Ki = 6.5 nM T31992 CSD29O 46237041 Ki = 682 nM T31992 CEB1X9 46237042 Ki = 6.9 nM T31992 C1VIK9 46237043 Ki = 66 nM T31992 C3RJ5M 46237044 Ki = 610 nM T31992 CU5Y9E 46237045 Ki = 70 nM T31992 CM7N6J 46237172 Ki = 62 nM T31992 CP15GJ 46237173 Ki = 78 nM T31992 CO2IU4 46704079 Ki = 149 nM T31992 CB85EQ 46704080 Ki = 92.3 nM T31992 CAE9Z3 46704081 Ki = 50.9 nM T31992 CD5V6T 46704082 Ki = 83.7 nM T31992 CNEO10 46871889 Ki = 112 nM T31992 C93AIR 46899573 Ki = 125000 nM T31992 CJ0R2O 46911381 Ki = 5.1 nM T31992 C03FQY 46943413 Ki = 118 nM T31992 C62ZDQ 51035422 Ki = 3.8 nM T31992 CW0CJ2 51035423 Ki = 6.5 nM T31992 CHF62Q 53361485 IC50 = 729 nM T31992 CJ3F4R 53361486 IC50 = 2440 nM T31992 C0NUM6 53386724 Ki = 7.7 nM T31992 C54FGU 53386866 Ki = 8.4 nM T31992 CRI54V 53386867 Ki = 4.9 nM T31992 CUX7S4 53386868 Ki = 14.6 nM T31992 CV40HR 53426278 Ki = 0.75 nM T31992 CCFP92 53516400 Ki = 7.9 nM T31992 C6SM5T 54613427 Ki = 87 nM T31992 CE2O3A 54768697 Ki = 76.4 nM T31992 C5SB4M 54768698 Ki = 80.6 nM T31992 CBNP25 54768699 Ki = 127 nM T31992 C9Z4RJ 54772055 Ki = 152 nM T31992 CB3EC8 54772057 Ki = 113 nM T31992 CE6LD4 54772059 Ki = 104 nM T31992 CD5P1I 54772061 Ki = 87.5 nM T31992 CK89GH 56659335 Ki = 7 nM T31992 C05JRQ 56659336 Ki = 8.9 nM T31992 CEC29W 56659337 Ki = 8.8 nM T31992 CZ4HI1 56662794 Ki = 7.4 nM T31992 CD8SR3 56662795 Ki = 27.7 nM T31992 CVM8W4 56666268 Ki = 7.2 nM T31992 C89SEG 56666269 Ki = 16.9 nM T31992 C36TYE 56666270 Ki = 7.6 nM T31992 CI2R9B 56676517 Ki = 0.92 nM T31992 C9X7VM 56676518 Ki = 10.1 nM T31992 C2U1VF 56679839 Ki = 9.1 nM T31992 CEZ3F5 56683163 Ki = 583 nM T31992 C4LB1M 56683164 Ki = 72 nM T31992 CZS9V5 56683165 Ki = 77 nM T31992 CIJ9V0 56684131 Ki = 844 nM T31992 CH52DA 56921864 Ki = 2830 nM T31992 CTFL92 56928044 Ki = 8.9 nM T31992 CP7YR5 57345662 Ki = 48 nM T31992 C0S2YZ 57383964 Ki = 8.5 nM T31992 C97GHV 57383965 Ki = 7.8 nM T31992 C4XF9A 57384114 Ki = 7.9 nM T31992 CS76WU 57384115 Ki = 16 nM T31992 C0UBL5 57384116 Ki = 8 nM T31992 C16AGY 57384117 Ki = 8.2 nM T31992 CV4C7B 57390570 Ki = 53.9 nM T31992 CS5O2D 57390571 Ki = 7.7 nM T31992 C14VNC 57390572 Ki = 9.5 nM T31992 C09GQI 57392249 Ki = 8.3 nM T31992 CY81SU 57392250 Ki = 10.7 nM T31992 CMEV16 57392251 Ki = 8.7 nM T31992 C94YIX 57392252 Ki = 41 nM T31992 CDP3C2 57392352 Ki = 6.3 nM T31992 CM7S3H 57394009 Ki = 10.3 nM T31992 CHAF57 57394010 Ki = 10.5 nM T31992 CV7K9Y 57394771 Ki = 125 nM T31992 CM4SL9 57394772 Ki = 55 nM T31992 C1M0LS 57394809 Ki = 730 nM T31992 CJ5XK2 57395770 Ki = 8.8 nM T31992 CV6QX4 57395771 Ki = 8.7 nM T31992 CP9D5B 57395861 Ki = 8.3 nM T31992 CHG91B 57396529 Ki = 108 nM T31992 C9H4VS 57396530 Ki = 8.5 nM T31992 C6XD2O 57397549 Ki = 8.6 nM T31992 C64VIW 57397550 Ki = 10.6 nM T31992 CR30XN 57397648 Ki = 19.8 nM T31992 CRIU35 57398318 Ki = 8.6 nM T31992 CN6TU2 57398319 Ki = 8.4 nM T31992 C97OJM 57399231 Ki = 8.5 nM T31992 C7XAZ3 57399232 Ki = 9.1 nM T31992 CK24NA 57399233 Ki = 8 nM T31992 CQD65L 57401080 Ki = 6.8 nM T31992 C1SK7F 57401081 Ki = 8.6 nM T31992 CG3X4V 57401764 Ki = 44 nM T31992 C4V5KY 57402747 Ki = 126 nM T31992 CRU53E 57402748 Ki = 807 nM T31992 C52TUM 57402749 Ki = 8.6 nM T31992 CQ9ZG2 57402750 Ki = 8.5 nM T31992 CI3L9R 57402843 Ki = 7.9 nM T31992 CW10QX 57402844 Ki = 7.1 nM T31992 C80WTZ 57403496 Ki = 129 nM T31992 CDIM87 57403497 Ki = 9.8 nM T31992 CW1TU4 57412422 Ki = 8.6 nM T31992 CT4BV9 57412423 Ki = 51 nM T31992 C31NWX 57412424 Ki = 22.4 nM T31992 CD86ER 57412425 Ki = 17.9 nM T31992 CB94YU 57412426 Ki = 8.7 nM T31992 C2K8YJ 57412507 Ki = 8.6 nM T31992 CSF4V6 57412508 Ki = 8.7 nM T31992 CHAO86 57412509 Ki = 15.3 nM T31992 C3U6TH 57412510 Ki = 55.9 nM T31992 C40LOS 57412511 Ki = 5.2 nM T31992 CZ47VT 57412512 Ki = 6.7 nM T31992 C28WRD 57412600 Ki = 50.2 nM T31992 C2XPG5 57413583 Ki = 9.2 nM T31992 CM2AY7 57413584 Ki = 24.8 nM T31992 C01TQW 59079460 Ki = 0.41 nM T31992 CGF3W6 66586679 Ki = 850 nM T31992 CN84CU 66586879 Ki = 840 nM T31992 C2Y5KV 70682044 Ki = 103 nM T31992 CXJ16H 71450117 Ki = 715 nM T31992 CB8JA3 71455488 Ki = 548 nM T31992 C02UHX 71455489 Ki = 931 nM T31992 CICJ97 71457274 Ki = 797 nM T31992 CMHG14 71521493 Ki = 5600 nM T31992 CHN53G 71521494 Ki = 4600 nM T31992 CZJ5M6 71521495 Ki = 2300 nM T31992 CFBE53 71521496 Ki = 4300 nM T31992 CME27W 71521497 Ki > 100000 nM T31992 C24XWU 71521575 Ki = 5900 nM T31992 CJF68W 71521576 Ki > 100000 nM T31992 C19OIY 71579130 Ki = 740 nM T31992 CV0LU6 71602117 Ki = 330 nM T31992 C1OPS4 71658869 Ki = 220 nM T31992 CN2FZ3 71659103 Ki = 180 nM T31992 C7NMJ2 71714066 Ki = 7240 nM T31992 C5DEF6 71714067 Ki = 12500 nM T31992 C50LSJ 71714068 Ki = 2440 nM T31992 CG4I1X 71718239 Ki = 740 nM T31992 C0LYX1 71718858 Ki = 860 nM T31992 CM24ND 71719433 Ki = 830 nM T31992 CT3D5S 71719441 Ki = 710 nM T31992 CIU4L2 71720670 Ki = 810 nM T31992 C0FM1E 72202020 Ki = 7 nM T31992 CT41SJ 72202021 Ki = 160 nM T31992 CX4G0R 72204928 IC50 > 10000 nM T31992 CG9C6U 72204929 IC50 > 10000 nM T31992 C5A6XZ 72204930 IC50 > 10000 nM T31992 C0XZK4 72204931 IC50 > 10000 nM T31992 C6RY4X 72204933 IC50 > 10000 nM T31992 C4N5AB 72204934 IC50 > 10000 nM T31992 C3H2FZ 72205111 IC50 = 82 nM T31992 CQ0VX7 72205112 IC50 = 8807 nM T31992 CQ7TI1 72205113 IC50 = 5500 nM T31992 CPAW52 72205114 IC50 = 4422 nM T31992 C2LD3J 72205115 IC50 = 6123 nM T31992 CX82JD 72696463 Ki = 138 nM T31992 COCV73 72696591 Ki = 42 nM T31992 C5KHD7 72696592 Ki = 220 nM T31992 C4FBA6 72696593 Ki = 3290 nM T31992 CO1JM5 72696594 Ki = 214 nM T31992 CUF61Q 72696595 Ki = 126 nM T31992 CJB8R7 72792832 Ki = 256 nM T31992 C5F7DT 72792833 Ki = 119 nM T31992 CAC7J8 72792834 Ki = 176 nM T31992 CFS02B 72792835 Ki = 40.1 nM T31992 CF5LW1 72792901 Ki = 23.7 nM T31992 C42IFJ 72792902 Ki = 45.3 nM T31992 CRMF25 72792903 Ki = 78.4 nM T31992 C2G5SR 72792904 Ki = 67 nM T31992 C6DR9O 72792905 Ki = 137 nM T31992 CGF5O1 72792967 Ki = 452 nM T31992 CWH3N9 72792968 Ki = 10.9 nM T31992 C5DSF8 72792969 Ki = 35.6 nM T31992 C2K6UZ 72792970 Ki = 67.3 nM T31992 CGI8K5 72793036 Ki = 15.9 nM T31992 C8WO6Z 72793037 Ki = 44.5 nM T31992 C6OZ0L 72793038 Ki = 50.1 nM T31992 CDTQ64 72793039 Ki = 58.9 nM T31992 CY16FM 72793040 Ki = 76 nM T31992 CXQN80 72793101 Ki = 148 nM T31992 CJ19BH 72793102 Ki = 24.9 nM T31992 CO1JT3 73054728 Ki = 340 nM T31992 C76RBA 86298624 IC50 = 593 nM T31992 C93FKI 86298625 IC50 = 70 nM T31992 CVLU48 86298626 IC50 = 82 nM T31992 CIJ96H 90644155 IC50 = 898 nM T31992 CX7EW1 90644156 IC50 = 6050 nM T31992 CK5GZ4 90644157 IC50 = 6050 nM T31992 C7O1YN 90644158 IC50 = 516 nM T31992 CEN6C1 90644159 IC50 = 92 nM T31992 C8X9UZ 90644160 IC50 > 10000 nM T31992 CQF98O 91827503 Ki = 39 nM T31992 C3I6NV 91827505 Ki = 9.6 nM T31992 CW1P4E 91827506 Ki = 5.8 nM T31992 CE2OY1 91995964 Ki = 0.26 nM T31992 CX45AP 92044053 Ki = 12.8 nM T31992 CDGZ03 101879106 Ki = 65.8 nM T31992 CY6ER7 101879108 Ki = 59 nM T31992 CUR4V8 114816322 Ki = 6.3 nM T31992 C0D1SQ 118724328 Ki = 238.6 nM T31992 C89YTC 118724329 Ki = 344 nM T31992 CBT87C 118724330 Ki = 70.9 nM T31992 C49AWZ 118724331 Ki = 48.2 nM T31992 CN16RY 122189300 Ki = 58 nM T31992 CYN3T8 122189301 Ki = 7.2 nM T31992 CSW9D1 122189302 Ki = 65 nM T31992 C6USQ7 122189303 Ki = 61 nM T31992 CQ4X1G 122189304 Ki = 64 nM T31992 CH1N0C 122193189 Ki = 640 nM T31992 C19HVL 122193190 Ki = 600 nM T31992 C5TQJ1 122193251 Ki = 750 nM T31992 C8XCL0 122193252 Ki = 310 nM T31992 CH4IV8 122194771 Ki = 0.67 nM T31992 CQ7N0L 122194772 Ki = 0.34 nM T31992 CI5K2F 122194773 Ki = 13.8 nM T31992 CV51IU 122194774 Ki = 0.69 nM T31992 C7OFR6 122194775 Ki = 0.84 nM T31992 C81HNW 122194776 Ki = 0.77 nM T31992 C8J5QV 122194777 Ki = 16.3 nM T31992 CV1C9T 122194778 Ki = 6.7 nM T31992 CJC1W3 122194779 Ki = 0.42 nM T31992 CU1TV5 122194780 Ki = 4.6 nM T31992 C4C1BE 122194781 Ki = 4 nM T31992 CR9I5Q 122194782 Ki = 0.83 nM T31992 C8SVY4 122194783 Ki = 3.6 nM T31992 C7HT8B 122194784 Ki = 8.5 nM T31992 CW8P3R 122194785 Ki = 3.7 nM T31992 COAK34 122194786 Ki = 0.67 nM T31992 CV4GW7 126961712 Ki = 3.2 nM T31992 C0FD4E 126961713 Ki = 3.4 nM T31992 CS2K4U 127034999 Ki = 7.4 nM T31992 CFG39M 127035855 Ki = 8 nM T31992 C6MH2V 127035856 Ki = 22.7 nM T31992 CVO4B6 127035857 Ki = 7.3 nM T31992 CQC6P9 127035858 Ki = 7.5 nM T31992 C7YA3N 127035859 Ki = 6.1 nM T31992 CXZI89 127035860 Ki = 6.5 nM T31992 C5KLP8 127035861 Ki = 7.7 nM T31992 CL76JS 127037630 Ki = 7.8 nM T31992 CSJ3V0 127041732 Ki = 53.6 nM T31992 CG75VH 127041733 Ki = 31.4 nM T31992 CP40EB 127049242 Ki = 4.4 nM T31992 CLFB54 127049248 Ki = 6.8 nM T31992 CG17IO 127050812 Ki = 7.3 nM T31992 C8X6CY 127050822 Ki = 4.4 nM T31992 C4IA5N 127051119 Ki = 6.2 nM T31992 CRDQ30 127051120 Ki = 4.6 nM T31992 C5Y4DI 127051953 Ki = 4.6 nM T31992 CJT9W0 135393499 Ki = 46.9 nM T31992 CK8FP3 135393500 Ki = 52.5 nM T31992 CRL4V7 135393501 Ki = 15.2 nM T31992 C4KH2F 136138702 Ki = 46.9 nM T31992 C2Z7GO 137637071 Ki = 4010 nM T31992 CK6OW4 137638637 Ki = 2.4 nM T31992 C6V8ED 137638882 Ki = 4.3 nM T31992 C64JQN 137639095 Ki = 374 nM T31992 C6B0CQ 137641198 Ki = 346 nM T31992 CXD9A0 137647636 Ki = 2915 nM T31992 C4N1MP 137650156 Ki = 25.6 nM T31992 CSTP12 137651755 Ki = 1.7 nM T31992 C8YV5D 137659052 Ki = 3930 nM T31992 CRC92Y 137661359 Ki = 325 nM T31992 C1Z8KG 137661675 Ki = 3.3 nM T31992 CT2ZB0 155515980 Ki = 7.8 nM T31992 CO7P5W 155531268 Ki = 11 nM T31992 CD4K6H 155556521 Ki = 7.7 nM T31992 CDB8T4 155568445 Ki = 29.8 nM T31992 C1C2GI 155569076 Ki = 53.7 nM T31992 D00FGB 11414131 Ki = 675 nM T31992 D00IAE 11974340 Ki = 83 nM T31992 D00IUB 13019 Ki = 29100 nM T31992 D00RNZ 910172 Ki = 5600 nM T31992 D00XIB 11680415 Ki = 842 nM T31992 D00XJA 711717 Ki = 3200 nM T31992 D00YEF 148885 Ki = 852 nM T31992 D01BUB 94952 Ki = 34000 nM T31992 D01OTW 46703932 Ki = 140 nM T31992 D01STY 9861037 Ki = 79 nM T31992 D01XFH 11851424 Ki = 11.3 nM T31992 D02BMV 46907399 Ki = 56.4 nM T31992 D02DBP 5054 Ki = 10700 nM T31992 D02QGI 273 Ki = 500 nM T31992 D03DAM 2725651 Ki = 730 nM T31992 D03KRB 45028567 Ki = 160 nM T31992 D03NBX 637308 Ki = 720 nM T31992 D03ZMQ 323 Ki = 48 nM T31992 D04CVC 4687472 Ki = 180 nM T31992 D04NSN 169682 Ki = 2900 nM T31992 D04VSP 46703768 Ki = 52.2 nM T31992 D05ETN 46703923 Ki = 70 nM T31992 D05JAJ 45028568 Ki = 59.7 nM T31992 D05QUG 45485279 Ki = 8400 nM T31992 D05TLB 11117301 Ki = 390 nM T31992 D05WQF 637540 Ki > 1000000 nM T31992 D05XZM 10081162 Ki = 3840 nM T31992 D06DYP 234562 Ki = 48 nM T31992 D06IOI 901953 Ki = 68.2 nM T31992 D07CYN 20347846 Ki = 5.8 nM T31992 D07LYW 11537386 Ki = 658 nM T31992 D07MTM 403 Ki = 10100 nM T31992 D07PNA 11660633 Ki = 2.2 nM T31992 D07QJJ 289 Ki = 48900 nM T31992 D07TAJ 914298 Ki = 6100 nM T31992 D08AOA 11543564 Ki = 61 nM T31992 D09JPC 16402 Ki = 640 nM T31992 D09PWX 8739 Ki = 780 nM T31992 D09TES 44395768 Ki = 68 nM T31992 D09TKG 25044690 Ki = 143 nM T31992 D09USO 5277466 IC50 = 309 nM T31992 D09WSJ 19772348 Ki = 711 nM T31992 D09WVV 8111 Ki = 10100 nM T31992 D0A0YX 5143 Ki = 773 nM T31992 D0A1CM 5281855 Ki = 8910 nM T31992 D0A6HS 6852129 Ki = 48 nM T31992 D0A8HW 44395685 Ki = 2.7 nM T31992 D0AU0M 637542 Ki = 6680 nM T31992 D0C4QB 44395769 Ki = 82 nM T31992 D0D4OV 20043772 Ki = 605 nM T31992 D0D6UR 12394434 Ki = 7800 nM T31992 D0E8CC 18794 Ki = 33 nM T31992 D0EJ9B 66827 Ki > 50000 nM T31992 D0G3BI 25090 Ki = 8600 nM T31992 D0G9NE 11659798 Ki = 341 nM T31992 D0H3NS 10752 Ki = 8200 nM T31992 D0HN0R 11623958 Ki = 48 nM T31992 D0J2AE 7377 Ki = 4800 nM T31992 D0J3SP 11718391 Ki = 24 nM T31992 D0J7GU 46703929 Ki = 98.3 nM T31992 D0KZ2D 11638641 Ki = 251 nM T31992 D0L5TZ 20195365 Ki = 6200 nM T31992 D0LC0F 96876 Ki = 6.5 nM T31992 D0LJ5P 44457221 Ki = 63.9 nM T31992 D0LU4S 156219 Ki = 8700 nM T31992 D0M3PO 69561 Ki = 680 nM T31992 D0M6RM 7365 Ki = 84000 nM T31992 D0N1AW 45485270 Ki = 46 nM T31992 D0NN3Q 78105 Ki = 1450 nM T31992 D0O0UE 729977 Ki = 46 nM T31992 D0O4KL 11640067 Ki = 7.3 nM T31992 D0O8WV 11536481 Ki = 5 nM T31992 D0OI1H 72894 Ki = 6500 nM T31992 D0OT5L 1631814 Ki = 8600 nM T31992 D0P6AM 3526523 Ki = 15 nM T31992 D0Q5VB 46704078 Ki = 95.7 nM T31992 D0Q7DJ 10742 Ki = 9140 nM T31992 D0R4KQ 46704077 Ki = 152 nM T31992 D0RB0D 44268050 Ki = 8800 nM T31992 D0SF3B 11529486 Ki = 40 nM T31992 D0T3NP 7456 Ki = 4100 nM T31992 D0TY8X 31036 Ki = 89 nM T31992 D0U4BB 10748 Ki = 9000 nM T31992 D0UM1I 12554666 Ki = 93.4 nM T31992 D0V5OW 46907400 Ki = 142 nM T31992 D0V9EN 689043 Ki = 8710 nM T31992 D0VD7H 84724 Ki = 280 nM T31992 D0W1OR 7424 Ki = 650 nM T31992 D0X5HL 15107 Ki = 590 nM T31992 D0Y3TZ 370 Ki = 7030 nM T31992 D0YU8J 1502014 Ki = 21 nM T31992 D0Z1HY 67136 Ki = 570 nM T73476 CZ17HE 445157 IC50 = 570 nM T73476 C62PJS 25114330 IC50 > 3000000 nM T73476 C5G3WD 25114332 IC50 > 1000000 nM T73476 C03IMY 46216724 IC50 > 300000 nM T73476 CZB9H4 46216725 IC50 > 300000 nM T73476 CEO59P 46231363 IC50 > 300000 nM T73476 C0R7FE 46231364 IC50 > 300000 nM T73476 CI2Q9S 46231365 IC50 > 300000 nM T73476 C3Y0ZF 46231366 IC50 > 3000000 nM T73476 CTJ7M6 46231367 IC50 > 1000000 nM T73476 CQL8T5 46231408 IC50 > 300000 nM T73476 CNGE41 46232215 IC50 > 300000 nM T73476 CW83FO 46232293 IC50 > 3000000 nM T73476 C9OM5J 46232294 IC50 > 3000000 nM T73476 CG5P2S 46232295 IC50 > 300000 nM T73476 CYCT81 46232296 IC50 > 1000000 nM T98711 D04AIT 5280445 Ki = 166100 nM T98711 D06OMW 3052776 IC50 = 4760 nM T98711 D06XWB 854026 IC50 > 100000 nM T98711 D07XYV 54766 IC50 = 3 nM T98711 D08USJ 4456 IC50 = 16300 nM T98711 D09QDP 4380 IC50 > 500000 nM T98711 D09QEI 4740 IC50 > 50000 nM T98711 D0B3HD 2519 IC50 > 50000 nM T98711 D0E6YQ 1935 IC50 = 0.9 nM T98711 D0K8KX 5280343 Ki = 68000 nM T98711 D0L4JT 5333 IC50 = 138790 nM T98711 D0NS6H 3152 IC50 = 14 nM T98711 D0O2WB 4991 IC50 = 900 nM T98711 D0Q0RC 3290 Ki = 20 nM T98711 D0R1QE 3672 IC50 < 600000 nM T98711 D0R9VR 9651 IC50 = 0.38 ug.mL-1 T98711 D0S2UG 26757 IC50 > 500000 nM T98711 D0UU9Y 4938 IC50 > 50000 nM T98711 D0W8WB 2353 IC50 = 1090 nM T98711 D0WY5Q 77991 IC50 = 30 nM T98711 D01LYX 65872 IC50 = 0.69 nM T98711 D02EVF 6112 IC50 > 1000000 nM T98711 D07CIN 192706 IC50 = 1560 nM T98711 D07SDQ 969516 IC50 > 5000 nM T98711 D0B1FE 3194 IC50 = 4600 nM T98711 D0B6IZ 137905 Ki > 100000 nM T98711 D0M3IN 1188 IC50 > 50000 nM T98711 D0U3EP 445154 IC50 > 5000 nM T98711 D09JVV 5983 IC50 = 15 nM T98711 D0B2BQ 135462830 IC50 = 7200 nM T98711 D0S1VV 119053 IC50 = 21000 nM T98711 CXU4W0 650 Ki > 100000 nM T98711 CT6RA0 2317 IC50 = 6165.95 nM T98711 C0RFA2 3102 Ki > 100000 nM T98711 C8F5QC 5077 IC50 = 11000 nM T98711 C8GZO5 5741 IC50 = 7273 nM T98711 CKB56J 5824 IC50 = 60 nM T98711 CX82HQ 6070 IC50 = 19460 nM T98711 C4IU5T 6889 Ki > 100000 nM T98711 C5NIV3 7088 IC50 = 19200 nM T98711 C5EUF4 7108 IC50 = 5800 nM T98711 C6NQ4X 8246 IC50 = 800 nM T98711 CJL02I 8307 IC50 = 1370000 nM T98711 CTY1W5 9820 Ki = 50 nM T98711 C25CYL 10434 Ki > 100000 nM T98711 C47FYB 10662 Ki > 100000 nM T98711 C2G5AW 11066 IC50 = 68000 nM T98711 COGY52 11321 Ki > 100000 nM T98711 C7U0TW 11747 Ki > 100000 nM T98711 C53FYO 11840 Ki > 100000 nM T98711 CKR3L9 12116 Ki > 100000 nM T98711 CU5KZ0 13005 Ki > 100000 nM T98711 CJ2GH1 13006 Ki > 100000 nM T98711 CG1LI5 14313 Ki > 100000 nM T98711 C4FW7E 18475 Ki > 100000 nM T98711 CTE5Z9 22006 IC50 = 14 nM T98711 C7S3JO 26257 Ki > 100000 nM T98711 C38JQX 31261 Ki > 100000 nM T98711 CN8A2G 38296 Ki > 100000 nM T98711 C7HE8W 38333 Ki > 100000 nM T98711 C0VK3I 39834 Ki > 100000 nM T98711 CVS6A8 40634 IC50 > 1000000 nM T98711 C8Z6TM 43402 Ki > 100000 nM T98711 CM94KL 47020 IC50 = 18000 nM T98711 CUNJ73 61209 Ki > 100000 nM T98711 C6U7FB 62539 Ki > 100000 nM T98711 C49ODY 65735 Ki = 610 nM T98711 C54XNY 68261 IC50 = 25100 nM T98711 C27NHT 69147 Ki > 100000 nM T98711 CN0ID1 69282 Ki > 100000 nM T98711 CW54JA 69288 Ki > 100000 nM T98711 C6BEN0 70945 Ki > 100000 nM T98711 C5KW4H 72311 IC50 = 10340 nM T98711 C2I7WP 74721 IC50 = 12000 nM T98711 CV8R4B 76561 Ki > 100000 nM T98711 CVJ78Y 79690 Ki > 100000 nM T98711 CAPG58 87502 Ki > 100000 nM T98711 C0EH3Z 88695 Ki > 100000 nM T98711 C70KGR 92036 Ki > 100000 nM T98711 C13IQL 93772 Ki > 100000 nM T98711 C8YU9Z 95415 Ki > 100000 nM T98711 CH91PI 95447 Ki > 100000 nM T98711 CAET12 101464 Ki = 90800 nM T98711 CR3E9L 103786 Ki > 100000 nM T98711 CG2VD5 120652 IC50 = 5248.07 nM T98711 CVB9H1 121587 IC50 > 50000 nM T98711 CVH8G6 122824 IC50 = 1600 nM T98711 C20LIY 136371 Ki > 100000 nM T98711 CTU83D 137777 Ki > 100000 nM T98711 CHAN02 138508 Ki > 100000 nM T98711 CYX5V0 142278 Ki > 100000 nM T98711 CF3I2J 156793 IC50 = 21770 nM T98711 C28RAT 165208 IC50 = 500 nM T98711 CIZE15 189688 IC50 > 100000 nM T98711 CX54PW 192442 IC50 = 3400 nM T98711 C5O8MF 197067 IC50 = 13680 nM T98711 C4VZL0 202767 IC50 > 1000000 nM T98711 C73HEY 203361 IC50 = 9800000 nM T98711 C1UW4K 204303 IC50 = 583000 nM T98711 CT8KV4 205772 IC50 = 52 nM T98711 C6W8MB 219592 Ki > 100000 nM T98711 COQ09W 219605 Ki > 100000 nM T98711 C25BHS 222475 Ki > 100000 nM T98711 CN35KE 222570 Ki > 100000 nM T98711 CP4W3S 229680 Ki > 100000 nM T98711 C0KV5M 236566 Ki > 100000 nM T98711 CE6U1D 237515 Ki > 100000 nM T98711 C92OSL 241331 Ki > 100000 nM T98711 C4N8IF 252525 IC50 > 30000 nM T98711 CHP1J7 262695 Ki > 100000 nM T98711 CDL3E1 262696 Ki > 100000 nM T98711 C6PU5E 270291 IC50 = 1570 nM T98711 CF62QN 275182 IC50 > 100000 nM T98711 C4HQ7V 284016 IC50 = 61010 nM T98711 CBR3Z7 302171 IC50 = 41300 nM T98711 CCSF19 303539 IC50 = 3026 nM T98711 C08WNV 317405 IC50 = 46770 nM T98711 CTMV50 321195 IC50 = 60000 nM T98711 CJ8RQ0 335358 IC50 = 1365 nM T98711 C5EI4Q 354120 Ki = 920 nM T98711 C5YJ7Z 359278 IC50 = 32 nM T98711 CHL04T 362574 IC50 = 800 nM T98711 CKS3U9 366710 Ki > 100000 nM T98711 C35JHV 385410 IC50 = 10320000 nM T98711 C5V0SH 386338 IC50 > 10000 nM T98711 C54EGJ 402658 IC50 = 26400 nM T98711 C9E5NG 402660 IC50 = 3300 nM T98711 CGKY63 402662 IC50 = 2300 nM T98711 CDCN80 402664 IC50 = 6700 nM T98711 C34VZP 402665 IC50 > 100000 nM T98711 C98AUK 402666 IC50 = 36000 nM T98711 C2SD4E 405589 IC50 > 50000 nM T98711 C7NU8P 409398 Ki = 17100 nM T98711 C5SFM6 412865 IC50 = 987 nM T98711 C18OIX 441064 IC50 > 100000 nM T98711 CLD6J9 441074 IC50 = 1230 nM T98711 CRN10Y 442113 IC50 = 4 nM T98711 CO9W4L 442854 IC50 = 35000 nM T98711 CE7GQ5 460616 IC50 = 1200 nM T98711 CQ3B5U 468188 IC50 = 5000 nM T98711 CU8GI1 468192 IC50 = 1100 nM T98711 CYMH94 471008 IC50 > 200000 nM T98711 CMO53J 475411 IC50 > 200000 nM T98711 C7U6FE 496015 IC50 = 2590 nM T98711 C0MI1O 513223 IC50 = 36000 nM T98711 CQ2F1V 513225 IC50 > 50000 nM T98711 CRI95J 513235 IC50 = 4200 nM T98711 CTWM69 586418 Ki > 100000 nM T98711 CH1E7N 590628 Ki > 100000 nM T98711 CCJQ96 599378 Ki > 100000 nM T98711 CL5E6W 607775 IC50 > 10000 nM T98711 CQ2M9X 638277 IC50 = 13000 nM T98711 CN71BS 641819 IC50 = 42000 nM T98711 C9MC2E 657348 IC50 = 16 nM T98711 C9CL3E 662730 IC50 = 6030 nM T98711 CVSQ83 662866 IC50 = 781 nM T98711 CXIK27 667496 IC50 = 3130 nM T98711 CK5V3P 667498 IC50 = 2490 nM T98711 CR1E5K 667801 IC50 = 25500 nM T98711 CJG47Q 704266 Ki = 190 nM T98711 C3DPV8 705751 Ki = 35000 nM T98711 CQP4B1 705773 Ki = 560 nM T98711 CFL0Y1 719823 IC50 = 49580 nM T98711 C9GU2E 744392 Ki = 23400 nM T98711 C50NVY 784043 IC50 = 3900 nM T98711 C4TAX6 784405 IC50 = 4000 nM T98711 C7PO1F 787366 IC50 = 7700 nM T98711 CO6AH8 806726 Ki = 9630 nM T98711 CB3GD4 818016 Ki = 4894000 nM T98711 CI8K6W 818170 IC50 = 56450 nM T98711 C29EOV 830741 IC50 = 9300 nM T98711 CMSC64 854531 IC50 > 10000 nM T98711 C5E3VW 866335 IC50 = 4920 nM T98711 CI54UD 866337 IC50 = 1090 nM T98711 C4BI6D 927411 IC50 > 50000 nM T98711 CA4D9I 931706 IC50 = 9820 nM T98711 CD3V9G 938070 IC50 = 61550 nM T98711 C84UPO 1018444 IC50 > 50000 nM T98711 C1YHE8 1208238 IC50 = 16600 nM T98711 CE7QJ6 1234089 IC50 = 51340 nM T98711 CYXQ78 1234090 IC50 = 37920 nM T98711 CED67Q 1237217 Ki = 1500 nM T98711 CC8JS7 1241150 IC50 = 42600 nM T98711 C3ZT7O 1320633 Ki = 6910 nM T98711 CM0I1K 1371037 Ki = 23000 nM T98711 CR37OY 1489313 IC50 = 250000 nM T98711 CIK9V0 1593398 IC50 = 83 nM T98711 CWTV42 1713189 Ki = 21000 nM T98711 C0EX9G 1755771 Ki > 100000 nM T98711 CB0ZP3 1812008 Ki > 100000 nM T98711 C9HL7Z 1816914 IC50 = 54090 nM T98711 CL8YK1 1889619 Ki = 90 nM T98711 C3FQD8 1906162 Ki > 100000 nM T98711 C3O6MN 1972026 Ki > 100000 nM T98711 C3X7MN 1991974 Ki = 20500 nM T98711 CI6ZU8 2133593 IC50 > 100000 nM T98711 CF37ZA 2147394 Ki > 100000 nM T98711 C0BEM3 2175773 IC50 > 50000 nM T98711 CJD8B3 2305233 Ki = 18100 nM T98711 CC5LI4 2326820 Ki = 2700 nM T98711 CN4U9J 2359994 IC50 = 5300 nM T98711 CC5J8U 2723754 IC50 = 23 nM T98711 CM6O4Z 2728673 IC50 = 57000 nM T98711 C68EBY 2728674 IC50 = 14000 nM T98711 C0OZQ2 2731126 Ki > 100000 nM T98711 CNKV06 2731127 Ki = 2390 nM T98711 CEM2C8 2731732 Ki > 100000 nM T98711 C2HOC5 2731733 Ki = 12300 nM T98711 CVC36I 2731902 Ki = 18900 nM T98711 CG62CN 2731904 Ki = 7400 nM T98711 CBEC45 2742082 IC50 > 30000 nM T98711 CN3KA4 2743222 IC50 < 10 nM T98711 C9R5LQ 2749125 Ki > 100000 nM T98711 C84DSN 2749126 Ki > 100000 nM T98711 CXU2J0 2755571 IC50 = 68000 nM T98711 C84VWR 2784639 Ki > 100000 nM T98711 CDCB42 2786143 Ki > 100000 nM T98711 C2RDM5 2886084 IC50 > 50000 nM T98711 CIK19R 2891624 IC50 = 443 nM T98711 CC8TY5 2915015 Ki = 7860 nM T98711 C6YQW9 2915964 Ki = 29100 nM T98711 CW9O2K 2930014 IC50 = 4.9 nM T98711 CRQ94D 2999234 IC50 > 100000 nM T98711 C1BM9V 3001811 IC50 > 200000 nM T98711 CC4OL6 3004425 Ki = 2150 nM T98711 CDR2K0 3012524 IC50 = 13880 nM T98711 C9QOY1 3029941 Ki = 510 nM T98711 CNYW30 3036637 IC50 = 529000 nM T98711 C04THC 3037884 IC50 = 1970 nM T98711 CZVE24 3041340 IC50 = 130000 nM T98711 C0JO2G 3055247 IC50 = 2400 nM T98711 CVN73X 3071771 IC50 = 25 nM T98711 CS5ET2 3071772 IC50 = 4100 nM T98711 CG09EQ 3071773 IC50 = 3100 nM T98711 CP2Y7N 3071774 IC50 = 3600 nM T98711 CZ6BA1 3071775 IC50 = 2900 nM T98711 C9M5PQ 3071776 IC50 = 1900 nM T98711 CI9VN7 3071777 IC50 = 1900 nM T98711 CC6W7T 3071778 IC50 = 1000 nM T98711 CIKF06 3071779 IC50 = 2700 nM T98711 CL2HU7 3071780 IC50 = 1300 nM T98711 CC9S8H 3072501 IC50 = 1800 nM T98711 CBLG95 3072502 IC50 = 3800 nM T98711 CS3L6G 3072503 IC50 = 3300 nM T98711 CIW2K3 3072504 IC50 = 2400 nM T98711 C2KN6J 3072505 IC50 = 3300 nM T98711 CEU74K 3072506 IC50 = 3800 nM T98711 CC56GR 3072507 IC50 = 1400 nM T98711 C4PCM1 3072508 IC50 = 4700 nM T98711 CHD8L0 3072509 IC50 = 6100 nM T98711 CU61MK 3072510 IC50 = 1300 nM T98711 CS1I6C 3072512 IC50 = 8400 nM T98711 CU20TQ 3072513 IC50 = 1600 nM T98711 C3KTC4 3072514 IC50 = 1100 nM T98711 C6QM9J 3072515 IC50 = 1800 nM T98711 CXLH39 3072518 IC50 = 5200 nM T98711 COW6E8 3075612 IC50 = 190 nM T98711 CU9Z2X 3083559 IC50 = 3000 nM T98711 CN5Z4H 3084319 IC50 = 2 nM T98711 CHEA42 3088389 IC50 = 4300 nM T98711 C1AM0S 3114312 Ki = 6710 nM T98711 C61RSW 3126152 Ki > 100000 nM T98711 CCP07Y 3264931 Ki > 100000 nM T98711 CB21VL 3321360 Ki > 100000 nM T98711 CZV6G2 3329233 Ki > 100000 nM T98711 C6NH9P 3469206 Ki > 100000 nM T98711 C3BT1N 3478673 IC50 = 45000 nM T98711 C10GCK 3527426 Ki > 100000 nM T98711 C3T1CV 3531512 Ki = 98900 nM T98711 CY6A2H 3706065 IC50 = 62000 nM T98711 CBZ13K 3722393 IC50 = 55800 nM T98711 C7V5YL 3748227 IC50 = 12200 nM T98711 CN5TX0 3756584 IC50 > 20000 nM T98711 CFV75H 3787603 IC50 = 4760 nM T98711 CV83OP 3796877 IC50 = 64800 nM T98711 C5UM2D 3821945 Ki > 100000 nM T98711 CU17BR 4088910 Ki > 100000 nM T98711 CR2X0V 4244497 Ki = 4690 nM T98711 CC1GF9 4338240 Ki > 100000 nM T98711 C8KV7I 4350924 Ki > 100000 nM T98711 C0V6QI 4369935 Ki > 100000 nM T98711 C42FGN 4384851 Ki > 100000 nM T98711 C01JRU 4416990 IC50 = 9100 nM T98711 CN9C3V 4513067 Ki > 100000 nM T98711 CAOH69 4789430 IC50 > 30000 nM T98711 CK9AT5 4792504 IC50 = 14000 nM T98711 CDV3O6 4846969 IC50 = 3000 nM T98711 C9MY1I 4885038 IC50 = 120 nM T98711 C5NJ3A 5004413 Ki > 100000 nM T98711 CNMY06 5038499 Ki > 100000 nM T98711 CL69XS 5127299 IC50 = 762 nM T98711 C7A0CD 5152006 IC50 = 2000 nM T98711 C0D3PO 5281671 IC50 = 1700 nM T98711 C5LGJ1 5282362 IC50 > 500000 nM T98711 C73SJW 5318015 IC50 > 100000 nM T98711 C5S6GW 5367146 IC50 = 105000 nM T98711 C32RHP 5367166 IC50 = 32000 nM T98711 C8HQN1 5376026 IC50 > 10000 nM T98711 CAC70Q 5377323 IC50 = 32000 nM T98711 CP1DZ2 5383464 IC50 = 27000 nM T98711 C25YUO 5458190 IC50 = 3170 nM T98711 C71CMO 5459840 IC50 = 506 ug.mL-1 T98711 CH6DT9 5481958 IC50 = 1700 nM T98711 CC6IV0 5481968 IC50 = 1700 nM T98711 CH8AJ6 5481969 IC50 = 1700 nM T98711 CMOI48 5481973 IC50 = 1700 nM T98711 CP69QB 5702326 IC50 > 5000 nM T98711 C81LVR 5702328 IC50 > 5000 nM T98711 CP46OW 5713121 IC50 = 1600 nM T98711 CGHW32 5747382 IC50 = 5100 nM T98711 C9L6KZ 5919802 IC50 = 31590 nM T98711 CYP0F4 6145899 IC50 = 119000 nM T98711 CR67NI 6333010 IC50 = 10 nM T98711 CK2MJ6 6333011 IC50 = 40 nM T98711 C8SZQ4 6410685 IC50 = 10000 nM T98711 C16EFR 6479925 IC50 = 100 nM T98711 CIL06S 6486743 IC50 = 18800 nM T98711 CNB34I 6540271 IC50 = 0.77 nM T98711 CW93TX 6610268 IC50 = 2140 nM T98711 C6EFT0 6712920 IC50 = 222 nM T98711 CSCO59 7580042 IC50 = 26070 nM T98711 C7BZ0N 7945979 IC50 > 5000 nM T98711 C9L0JT 9574517 IC50 = 240 nM T98711 CSY0F8 9574537 IC50 > 50000 nM T98711 CCLX43 9579448 IC50 = 2600 nM T98711 CK37WV 9579449 IC50 > 50000 nM T98711 C8XKM7 9794806 IC50 = 100 nM T98711 CU2XN7 9819233 IC50 = 1560 nM T98711 CFHP83 9822470 IC50 = 1570 nM T98711 CVDM07 9828345 IC50 = 257 nM T98711 CG6W8R 9839754 IC50 = 920 nM T98711 C7C0IP 9843814 Ki = 1400 nM T98711 CM0BX3 9850331 IC50 = 164 nM T98711 CKA8W7 9851127 IC50 = 194 nM T98711 C4VHS5 9859456 IC50 = 3100 nM T98711 CF05ZV 9864626 IC50 = 51 nM T98711 C2NLZ5 9886877 IC50 = 28100 nM T98711 CME5I4 9894056 IC50 = 26 nM T98711 C94UJV 9905831 IC50 = 1560 nM T98711 CE8M7Y 9928503 Ki = 20 nM T98711 CE69LQ 9952812 IC50 > 10000 nM T98711 CFW16Y 9958700 IC50 = 132 nM T98711 CYLG46 9959612 IC50 = 5.66 nM T98711 CC3G7N 9961034 IC50 = 3.3 nM T98711 CP3QN4 9976101 IC50 = 4800 nM T98711 C2WYT7 9976761 IC50 = 3900 nM T98711 CFH1O0 9992823 IC50 = 6.8 nM T98711 CI3D7M 10038341 IC50 = 59.4 nM T98711 CH0R1M 10038557 IC50 > 50000 nM T98711 C30ZHN 10040889 IC50 = 4300 nM T98711 CN0HU2 10044997 IC50 = 155000 nM T98711 CI2X0Z 10075220 IC50 = 0.6 nM T98711 CEKX28 10094001 IC50 > 50000 nM T98711 CWD41K 10097011 IC50 = 13.9 nM T98711 CTI26V 10098048 IC50 > 200000 nM T98711 CI70JE 10109540 IC50 > 50000 nM T98711 C68RJB 10110147 IC50 = 9000 nM T98711 CTQ95J 10110914 IC50 = 4200 nM T98711 CVWT04 10117403 IC50 = 13650 nM T98711 CSX92P 10126521 IC50 > 50000 nM T98711 C1B9MQ 10150601 IC50 > 50000 nM T98711 CA5J4V 10150622 IC50 > 50000 nM T98711 CO6I2N 10159339 IC50 = 890 nM T98711 CMJ4S6 10161755 IC50 = 31550 nM T98711 CV65OE 10179120 IC50 = 780 nM T98711 CQB9D0 10200831 IC50 = 26700 nM T98711 CD0P4U 10204915 IC50 = 22190 nM T98711 CS9E7Y 10205836 IC50 = 15670 nM T98711 C36DNM 10215997 IC50 > 50000 nM T98711 CP1HT3 10223679 IC50 = 250 nM T98711 CX4Y1T 10224148 IC50 = 15230 nM T98711 CY6I8F 10243365 Ki = 685200 nM T98711 CWZ5S0 10245631 IC50 = 516 nM T98711 CU6B5G 10255032 IC50 = 4840 nM T98711 C81ONP 10255275 IC50 = 18000 nM T98711 C8MAO5 10268794 Ki = 210 nM T98711 CD89EN 10272949 IC50 = 10790 nM T98711 C3GMK4 10277339 IC50 = 38400 nM T98711 CM19RC 10277340 IC50 = 57870 nM T98711 C7ZIP3 10277830 IC50 = 23210 nM T98711 CB2K1F 10287897 IC50 > 50000 nM T98711 C0TWQ3 10292083 IC50 = 6200 nM T98711 C08TOG 10299954 IC50 = 26830 nM T98711 C72VTB 10300579 IC50 = 78920 nM T98711 CV5B1A 10308583 IC50 > 50000 nM T98711 CJ0VN5 10310052 IC50 > 50000 nM T98711 C7NRO3 10317909 IC50 = 75000 nM T98711 CPRK30 10337156 IC50 = 23500 nM T98711 C4Z7DT 10337617 IC50 = 300000 nM T98711 CGZ5B9 10342292 IC50 = 1700 nM T98711 C1VFO0 10355816 IC50 > 2000 nM T98711 CRI5E2 10360601 IC50 = 1 nM T98711 C3H0MY 10372514 IC50 = 2238.72 nM T98711 CC5WG8 10416369 IC50 = 4.9 nM T98711 CB0VE3 10458051 IC50 = 31200 nM T98711 CI7C9Y 10464995 IC50 > 10000 nM T98711 CFN3I9 10472189 IC50 = 101910 nM T98711 CU21VN 10476544 IC50 > 50000 nM T98711 CHM50O 10481357 IC50 = 10.4 nM T98711 C7J2KT 10502606 IC50 = 776 nM T98711 CK5W8X 10505674 IC50 = 641 nM T98711 CGH7U6 10526350 IC50 = 85800 nM T98711 CWUY91 10539341 IC50 = 18900 nM T98711 C98RWG 10545891 IC50 = 21.8 nM T98711 CM3UP4 10550262 IC50 = 91200 nM T98711 CJ0N1R 10569957 IC50 = 1589.5 nM T98711 CIS15A 10573780 IC50 = 85.3 nM T98711 CYSD36 10593041 IC50 = 1430 nM T98711 C3XYI4 10597848 IC50 = 7086 nM T98711 CVD9A1 10610498 IC50 = 237 nM T98711 CTM40A 10615903 IC50 = 1745.5 nM T98711 C2LRS9 10622407 IC50 = 600 nM T98711 CV1PG0 10623652 IC50 = 85 nM T98711 CY93KL 10625415 IC50 = 53 nM T98711 CWE41Q 10655805 Ki > 100000 nM T98711 CZ59MX 10663695 IC50 = 396 nM T98711 CL95NU 10664401 IC50 = 730 nM T98711 CSIC19 10690207 IC50 = 78 nM T98711 CNR15Z 10713570 IC50 = 340 nM T98711 CG4Z8N 10721720 IC50 = 0.69 nM T98711 CL1BE8 10729509 IC50 = 42000 nM T98711 CRD47N 10730136 IC50 = 1120.5 nM T98711 CT68IS 10757271 IC50 = 952 nM T98711 C4O5KP 10763156 IC50 = 43800 nM T98711 CDAR18 10764956 IC50 = 8.1 nM T98711 C2AN5S 10774819 IC50 = 5900 nM T98711 CFHV29 10778312 IC50 = 197 nM T98711 C9PTG2 10785532 IC50 = 310 nM T98711 C4YS9A 10789991 IC50 = 156270 nM T98711 C9YLN1 10799366 IC50 = 12200 nM T98711 CKZ53Y 10825928 IC50 = 81000 nM T98711 CD0L7C 10848598 IC50 > 2000 nM T98711 C8G6BS 10850978 IC50 = 46 nM T98711 CGL0K9 10855014 IC50 = 2511.89 nM T98711 C8XSW2 10863593 Ki = 16200 nM T98711 CHF26C 10872974 IC50 = 270 nM T98711 CF28NJ 10879668 Ki > 100000 nM T98711 C3HZ6S 10894911 IC50 = 510 nM T98711 C1PZ2V 10896395 IC50 = 16.5 nM T98711 CH49NV 10899196 Ki > 100000 nM T98711 CP93JE 10902085 Ki > 100000 nM T98711 C95XSO 10905408 IC50 = 280 nM T98711 CU4W9S 10909176 IC50 = 758.58 nM T98711 CV35KR 10909236 IC50 = 2570.4 nM T98711 CSW4G1 10915203 IC50 = 815 nM T98711 C4M3ZI 10919451 IC50 = 8317.64 nM T98711 CR19FE 10927360 IC50 = 25 nM T98711 C3DSY6 10927599 IC50 = 42.6 nM T98711 CCS2Y7 10941381 IC50 = 7413.1 nM T98711 C0I9NT 10943454 IC50 > 10000 nM T98711 CZSC17 10958661 IC50 > 10000 nM T98711 C2Y5XC 10961666 IC50 = 3650 nM T98711 C2WRK0 10963725 IC50 = 165.96 nM T98711 CK72HO 10974737 IC50 = 165958.69 nM T98711 CJ7DR2 10985959 IC50 = 7585.78 nM T98711 CQ4ZC5 10996738 IC50 = 1659.59 nM T98711 C4NY9F 11006704 IC50 = 3.9 nM T98711 CD96QS 11007082 IC50 = 54954.09 nM T98711 C7NZY9 11009341 Ki > 100000 nM T98711 C9PTO8 11027124 IC50 = 53700 nM T98711 C0F1HL 11027759 IC50 = 2000 nM T98711 CN6WF9 11051398 IC50 = 83.18 nM T98711 CO30RK 11081720 IC50 = 310600 nM T98711 CPSM68 11104192 IC50 = 2630.27 nM T98711 CSYM37 11104646 IC50 = 2137.96 nM T98711 CF15NS 11113449 Ki = 3400 nM T98711 CJ0RG8 11113852 Ki = 26300 nM T98711 CUZ1H3 11114008 IC50 > 30000 nM T98711 C74KUO 11115691 IC50 = 6456.54 nM T98711 CJ2P6K 11121264 IC50 > 10000 nM T98711 CST19B 11124861 IC50 = 7.5 nM T98711 CKJ49N 11125225 IC50 = 5495.41 nM T98711 CKRZ24 11125922 IC50 = 1412.54 nM T98711 C1Q5OP 11136870 IC50 = 2398.83 nM T98711 C7FPU3 11146640 IC50 = 1071.52 nM T98711 CIP41D 11150497 IC50 = 410 nM T98711 C8FNC1 11156231 IC50 = 0.03 nM T98711 C9LFS7 11156598 IC50 = 0.1 nM T98711 C7JC9B 11167725 IC50 = 16 nM T98711 CGWM68 11168014 IC50 = 206 nM T98711 C8UTA5 11169647 IC50 = 63.7 nM T98711 CYL18X 11179973 IC50 = 70300 nM T98711 C9IV7T 11181553 IC50 = 1621.81 nM T98711 C4EU7X 11188905 IC50 = 1000 nM T98711 C6L0IS 11190153 IC50 = 329 nM T98711 CZ2GU4 11191030 IC50 = 79 nM T98711 C3D5SL 11191634 IC50 = 3.4 nM T98711 CBJV46 11192468 IC50 = 40200 nM T98711 CM54US 11192952 IC50 = 84400 nM T98711 CSJ1R4 11193161 IC50 = 330 nM T98711 CH30SU 11204324 IC50 = 81300 nM T98711 CE21OG 11204682 IC50 = 15488.17 nM T98711 C9EMG6 11209350 IC50 = 2000 nM T98711 CZPB69 11210161 IC50 = 200 nM T98711 CJI9N3 11216927 IC50 = 1096.48 nM T98711 C7X9ZC 11221007 Ki = 860 nM T98711 C4N9ZL 11221206 IC50 = 100 nM T98711 C1NI8D 11222968 IC50 > 10000 nM T98711 CY86GP 11226206 IC50 = 44300 nM T98711 CX6CF4 11232205 IC50 = 130 nM T98711 CEXP98 11233503 IC50 = 27 nM T98711 CT38EP 11235216 IC50 > 50000 nM T98711 C6TVW3 11238481 IC50 = 500 nM T98711 CSXF65 11238662 IC50 = 610 nM T98711 CV73WE 11239040 IC50 = 761000 nM T98711 C5FO1B 11243200 IC50 = 370 nM T98711 C6GHQ3 11244670 IC50 = 14000 nM T98711 CRL20G 11249115 IC50 = 2.9 nM T98711 C8GJD2 11249560 IC50 = 5.7 nM T98711 C6LH1M 11250361 IC50 = 130000 nM T98711 C81GLD 11257074 IC50 = 8.3 nM T98711 CKTJ19 11260293 IC50 > 30000 nM T98711 CPSO84 11261638 IC50 = 9000 nM T98711 CP6FX1 11268904 IC50 = 900 nM T98711 CEBK83 11272051 IC50 = 22.4 nM T98711 CC14OZ 11272989 IC50 = 155000 nM T98711 CAP59Z 11278342 IC50 = 50 nM T98711 CYRB74 11283475 IC50 = 11.7 nM T98711 C2CQH5 11283831 IC50 = 4650000 nM T98711 C1JKX2 11290299 IC50 = 100 nM T98711 CE79LQ 11290672 IC50 = 2165 nM T98711 CXV91C 11304331 IC50 > 50000 nM T98711 CKD79X 11304963 IC50 = 47.5 nM T98711 CBL8D9 11314048 IC50 = 4000 nM T98711 C2SQ3D 11314386 IC50 > 50000 nM T98711 CX9JQ2 11316712 IC50 = 12 nM T98711 CAJ8O0 11316986 IC50 = 1 nM T98711 CEKG13 11329992 IC50 = 57900 nM T98711 C9JV3E 11330142 Ki = 8.59 nM T98711 CNTY27 11336871 IC50 = 460 nM T98711 C7RJ4Z 11341331 IC50 = 5.6 nM T98711 CG91BA 11350292 IC50 > 50000 nM T98711 CM34HL 11352229 IC50 = 3.24 nM T98711 CAR45P 11359651 IC50 = 900 nM T98711 C59YIW 11359764 IC50 = 24400 nM T98711 CK49FX 11364765 IC50 = 600 nM T98711 CSE62M 11365562 IC50 = 136000 nM T98711 CQU73N 11376655 IC50 = 40 nM T98711 CI0CV9 11378169 IC50 = 660.69 nM T98711 CIAR80 11380022 IC50 = 6 nM T98711 CPB6X4 11381434 IC50 > 10000 nM T98711 CFS5X7 11382561 IC50 = 10.4 nM T98711 CSDY73 11385572 IC50 = 5.04 nM T98711 C61VUW 11392125 IC50 = 4 nM T98711 CPNA70 11393196 IC50 > 30000 nM T98711 CJAL17 11397926 IC50 = 77 nM T98711 CWB6K1 11404631 IC50 = 416 nM T98711 C8W9AR 11409935 IC50 = 11.7 nM T98711 CR7E9T 11420352 IC50 = 5500 nM T98711 CXLY31 11425531 IC50 = 24 nM T98711 CL9G3Y 11425872 IC50 = 200 nM T98711 C7T8KU 11432076 IC50 = 3.2 nM T98711 C5DML9 11432727 IC50 = 600 nM T98711 C83YSD 11434003 IC50 = 95499.26 nM T98711 CY72LB 11438752 IC50 > 30000 nM T98711 CL15TO 11445385 IC50 = 8490 nM T98711 C5TOG0 11445610 IC50 = 2190 nM T98711 CS7U9F 11455392 IC50 = 21.4 nM T98711 CY3EG9 11457400 IC50 = 1862.09 nM T98711 CKU29D 11461464 IC50 = 612 nM T98711 CAE18Q 11464843 IC50 = 11400000 nM T98711 C2N7YB 11465667 IC50 = 1.7 nM T98711 CA92CF 11465956 IC50 = 19 nM T98711 C9E6RY 11478767 IC50 = 1.7 nM T98711 C1KBO3 11478903 IC50 = 94600 nM T98711 C19ONS 11482774 IC50 = 2 nM T98711 C3WVS4 11489952 Ki = 0.74 nM T98711 CFQ27V 11490183 IC50 = 400 nM T98711 CSQZ71 11495096 IC50 = 12 nM T98711 C7OR8M 11504245 IC50 = 3 nM T98711 C94WCH 11509353 IC50 = 1.09 nM T98711 CVN51A 11514475 IC50 = 3 nM T98711 CA07BP 11530167 IC50 = 5100 nM T98711 CHLC49 11539744 IC50 = 0.68 nM T98711 C4CA7T 11550697 IC50 = 120 nM T98711 CY9MU1 11563410 IC50 = 25 nM T98711 CPHO51 11566532 IC50 = 15 nM T98711 C9XNM6 11573923 IC50 = 54 nM T98711 CWI4A2 11574168 IC50 = 23 nM T98711 C6P0EV 11576166 IC50 = 20000 nM T98711 C48YEL 11581590 IC50 > 50000 nM T98711 CH04PB 11588880 IC50 = 0.87 nM T98711 C3WQI0 11595988 IC50 > 50000 nM T98711 C2C4KA 11599119 IC50 = 35 nM T98711 CK2PB1 11603489 IC50 = 0.25 nM T98711 CLOD63 11606144 IC50 = 23 nM T98711 COAU76 11620371 IC50 = 6.8 nM T98711 CSDF87 11624531 IC50 = 13 nM T98711 CAF5O0 11625278 IC50 = 0.89 nM T98711 C2LD0Q 11631221 IC50 = 52000 nM T98711 CV5RH1 11631680 IC50 = 1180 nM T98711 CMH6K9 11632307 IC50 = 5100 nM T98711 CEY1C7 11645534 IC50 = 11400 nM T98711 CQX1I8 11647230 IC50 = 82400 nM T98711 CBGT09 11648619 IC50 = 12.6 nM T98711 CAE18N 11653182 IC50 = 72 nM T98711 CU1K8W 11666118 IC50 = 28 nM T98711 C67HTG 11667904 IC50 > 50000 nM T98711 C27AHE 11668852 IC50 > 50000 nM T98711 C8E6NF 11669798 IC50 = 9.5 nM T98711 C0AR9Z 11681391 IC50 = 36400 nM T98711 CI5MT9 11681880 IC50 = 40 nM T98711 C47LNU 11682017 IC50 > 50000 nM T98711 CC1ZN6 11694595 IC50 = 23 nM T98711 CR1IW0 11697764 IC50 = 3600 nM T98711 C5HYV7 11698149 IC50 = 2490 nM T98711 CL41DM 11698541 IC50 > 50000 nM T98711 CJ6UR7 11706508 IC50 = 7.8 nM T98711 C71EWN 11713155 IC50 = 1 nM T98711 C5FJ0D 11722860 IC50 = 897 nM T98711 C45PDY 11734220 IC50 = 4000 nM T98711 CBY03I 11739675 IC50 = 22 nM T98711 C1SDF0 11752376 IC50 = 8.58 nM T98711 C51RYW 11752643 IC50 = 32 nM T98711 CLMV71 11753218 Ki = 3.13 nM T98711 CQB14T 11763573 IC50 = 153000 nM T98711 C7MFV8 11763757 IC50 = 18620.87 nM T98711 C7OPQ0 11772375 IC50 = 300 nM T98711 CV84AY 11776726 IC50 = 2.4 nM T98711 CV4W8C 11784091 IC50 = 480 nM T98711 CZRE80 11786613 IC50 = 100 nM T98711 CG34JX 11792247 IC50 = 1473 nM T98711 CQ6YH2 11799236 IC50 = 513 nM T98711 CS23AV 11800047 IC50 = 1.36 nM T98711 CCQN45 11805526 Ki > 100000 nM T98711 C7WYG3 11810853 IC50 = 1600 nM T98711 CX97ZV 11814517 IC50 = 4073.8 nM T98711 CVS5N8 11854653 IC50 = 1.7 nM T98711 CCH27V 12013999 IC50 = 18900 nM T98711 CTM34I 12109666 IC50 = 224670 nM T98711 CJC3N0 12146686 IC50 > 30000 nM T98711 CKG7A0 12222796 Ki > 100000 nM T98711 CC3MQ9 12314224 IC50 = 56 nM T98711 CD1J7E 12851056 Ki = 24700 nM T98711 C5L0GN 12927905 IC50 = 541000 nM T98711 C1R4MF 12995052 IC50 = 230 nM T98711 C54QHI 13006034 IC50 = 250 nM T98711 C6XHS1 13006035 IC50 = 1820 nM T98711 CG7AZ9 13006036 IC50 = 165 nM T98711 CDP08C 13006037 IC50 = 170 nM T98711 C0AH2N 13006038 IC50 = 66 nM T98711 CIY8G4 13006039 IC50 = 798 nM T98711 CTX5Q6 13006040 IC50 = 490 nM T98711 CJ43VT 13006041 IC50 > 10000 nM T98711 CS7V4K 13006042 IC50 = 5020 nM T98711 CT5C2K 13006043 IC50 = 3290 nM T98711 CH46IX 13006044 IC50 = 1100 nM T98711 C3VSW6 13006045 IC50 = 650 nM T98711 CFE3W8 13006046 IC50 = 3890 nM T98711 CU0BN1 13006047 IC50 = 8530 nM T98711 CAJG53 13300537 IC50 = 840000 nM T98711 C0KSR2 13497076 IC50 = 150000 nM T98711 CEO81S 13552185 IC50 = 1400000 nM T98711 CL4MK3 13552226 IC50 = 120000 nM T98711 C4TA0V 13735450 IC50 > 5000 nM T98711 C8B5LO 13780062 Ki > 100000 nM T98711 C3YOX2 13827082 Ki > 100000 nM T98711 C4CR1L 13827083 Ki > 100000 nM T98711 CK08BO 13896866 IC50 > 500000 nM T98711 C0TRN9 13934286 IC50 > 200000 nM T98711 CU2M9R 14107712 IC50 = 2489 nM T98711 C4YBN3 14109375 IC50 > 200000 nM T98711 CJS4R6 14193572 IC50 = 10 nM T98711 CM6R4N 14193573 IC50 = 3 nM T98711 C39VGI 14193575 IC50 = 3 nM T98711 C6BP1S 14193577 IC50 = 2 nM T98711 C0PO5M 14349781 IC50 = 290 nM T98711 CJZ46W 14353465 IC50 = 3570 nM T98711 C7NE3Y 14372818 IC50 = 41 nM T98711 CQA53V 14537189 Ki = 1300 nM T98711 CX7AE6 14537192 Ki = 800 nM T98711 CD0F5X 14537193 Ki = 4600 nM T98711 CTB5H2 14539882 IC50 = 1700 nM T98711 CULX32 14553493 IC50 = 1670 nM T98711 CH27JR 14609844 IC50 = 7883 nM T98711 C93MXE 14735915 IC50 = 53000 nM T98711 CAH47C 14735925 IC50 = 34000 nM T98711 CMF7U1 14877070 IC50 = 140000 nM T98711 CK69GO 15005009 IC50 = 18000 nM T98711 C6V9HJ 15005010 IC50 = 1100 nM T98711 C1EQ0S 15043261 IC50 = 17990 nM T98711 C8PYV9 15043264 IC50 = 18200 nM T98711 CL2C7Y 15044210 Ki > 100000 nM T98711 CNJ2A9 15085436 IC50 = 71 nM T98711 CJ3E7T 15125273 IC50 = 690 nM T98711 CA13LZ 15125274 IC50 = 4230 nM T98711 C9WTF1 15125278 IC50 = 2070 nM T98711 CVJP83 15289585 IC50 > 1000000 nM T98711 CZ3WJ2 15490813 IC50 = 273 nM T98711 C1S6GM 15720175 IC50 = 17 nM T98711 CR2J0F 16094841 IC50 = 12.1 nM T98711 C34FJR 16094854 IC50 = 12.8 nM T98711 C8JM2I 16094855 IC50 = 7.13 nM T98711 CCL15D 16094856 IC50 = 0.969 nM T98711 COID78 16094857 IC50 = 0.293 nM T98711 CMT73Z 16094858 IC50 = 6.03 nM T98711 C3RN7X 16094859 IC50 = 0.226 nM T98711 CWI3K1 16094860 IC50 = 0.141 nM T98711 CG14KR 16094871 IC50 = 27.6 nM T98711 CKJ3F6 16094872 IC50 = 1.68 nM T98711 CD9S2E 16094873 IC50 = 0.523 nM T98711 C35HXC 16094875 IC50 = 24 nM T98711 CU8W5V 16094876 IC50 = 0.139 nM T98711 CMKY94 16114893 IC50 > 50000 nM T98711 C9E6AH 16114898 IC50 > 50000 nM T98711 C4RCO2 16115141 IC50 > 50000 nM T98711 C28IBN 16219608 IC50 = 420 nM T98711 C6GD9H 16235993 IC50 > 5000 nM T98711 CFX56U 16407549 IC50 = 270 nM T98711 CG5J7B 16584800 IC50 = 214410 nM T98711 C6K4AZ 16645662 Ki = 45400 nM T98711 C7MSU0 16653132 IC50 > 100000 nM T98711 C1JKF6 16664256 IC50 = 555500 nM T98711 CH9Y5B 17159064 IC50 = 3500 nM T98711 C5ZMI9 17159212 IC50 = 7200 nM T98711 CF6ZW1 17159244 IC50 = 11000 nM T98711 C80YMT 17159252 IC50 = 7800 nM T98711 CL2IW7 17422256 IC50 = 1360 nM T98711 CM9AH0 17602492 IC50 = 10300 nM T98711 C91BCT 17652420 Ki = 42500 nM T98711 C2OF8S 18471933 Ki > 100000 nM T98711 CFD89G 18870980 IC50 = 656850 nM T98711 C2QZ4O 18870983 IC50 = 11020 nM T98711 C39VUS 19760985 IC50 = 10420 nM T98711 CW0H1Y 20055993 IC50 > 200000 nM T98711 CU5Y8N 20208765 IC50 = 61659.5 nM T98711 C0Q9VM 20208772 IC50 = 13803.84 nM T98711 C45TLN 21204337 IC50 = 51000 nM T98711 C0ET8M 21362734 IC50 > 10000 nM T98711 C72BMS 21409569 IC50 = 22700 nM T98711 CQKH16 21592283 IC50 = 188360 nM T98711 CJKR07 21632954 IC50 > 200000 nM T98711 CEJ49C 21633084 IC50 > 200000 nM T98711 C2FBA3 21672659 IC50 > 30000 nM T98711 CX8W6N 21839636 IC50 = 63.3 nM T98711 CT3YN1 21839638 IC50 = 543 nM T98711 C5GZ1L 21839640 IC50 = 32.4 nM T98711 C8YO3H 21839642 IC50 = 109 nM T98711 CWR90B 21839649 IC50 = 89 nM T98711 CI29XS 22064898 IC50 > 100000 nM T98711 CYUW32 22181436 IC50 = 36800 nM T98711 C1DL8N 22210859 IC50 = 570 nM T98711 CYF5N8 22210860 IC50 = 27000 nM T98711 CYQB56 22210861 IC50 = 26000 nM T98711 C10ZWQ 22210862 IC50 = 3900 nM T98711 CH5YQ0 22210863 IC50 = 1800 nM T98711 CM3Y1I 22574246 Ki > 100000 nM T98711 C5IZQ8 23093594 IC50 = 1400 nM T98711 CHO5K2 23102336 Ki = 150 nM T98711 C7KCD5 23247894 IC50 > 200000 nM T98711 CZ0L4G 23277102 IC50 = 46000 nM T98711 CK15SO 23448959 IC50 = 38600 nM T98711 C13RZX 23624871 IC50 = 505 nM T98711 CZ7ET2 23634635 IC50 > 10000 nM T98711 CQ91XS 23634752 IC50 > 10000 nM T98711 CSK7Z4 23634753 IC50 > 10000 nM T98711 COZ1U3 23634754 IC50 > 10000 nM T98711 CIR09L 23634873 IC50 > 10000 nM T98711 CJMI97 23634874 IC50 = 375 nM T98711 CO5D8M 23634876 IC50 = 1450 nM T98711 CNFK89 23635382 IC50 > 10000 nM T98711 C0LA7S 23635383 IC50 > 10000 nM T98711 C15ASX 23635398 IC50 > 50000 nM T98711 C9F1MQ 23635399 IC50 > 50000 nM T98711 CXIA45 23635400 IC50 > 50000 nM T98711 CQ0H4M 23635401 IC50 > 50000 nM T98711 CZ5R6B 23635511 IC50 > 50000 nM T98711 C5S2QB 23635512 IC50 > 50000 nM T98711 C4B8MX 23635513 IC50 > 50000 nM T98711 CWD7J8 23635514 IC50 > 50000 nM T98711 C0ASM1 23635515 IC50 > 50000 nM T98711 CKP70J 23635516 IC50 > 50000 nM T98711 CM0X3T 23635632 IC50 > 50000 nM T98711 C0VL9W 23635633 IC50 > 50000 nM T98711 CJ73KM 23635634 IC50 > 50000 nM T98711 CWI26H 23635635 IC50 > 50000 nM T98711 CP6J2G 23635636 IC50 > 50000 nM T98711 C4GA2J 23635637 IC50 > 50000 nM T98711 CTJ96S 23635746 IC50 > 10000 nM T98711 C1P7GL 23635748 IC50 > 10000 nM T98711 CV8QU5 23635749 IC50 > 10000 nM T98711 CT46CR 23635766 IC50 = 19000 nM T98711 CVJ6C0 23635767 IC50 > 50000 nM T98711 CU61DC 23635768 IC50 > 50000 nM T98711 C74DZC 23635875 IC50 = 1535 nM T98711 CGJ6U3 23635876 IC50 = 380 nM T98711 CF91IH 23635891 IC50 > 50000 nM T98711 CT67MK 23635892 IC50 > 50000 nM T98711 CKM0C8 23635893 IC50 > 50000 nM T98711 CC1PX4 23635894 IC50 > 50000 nM T98711 C0XQ8E 23635895 IC50 = 8200 nM T98711 CCPS26 23635896 IC50 > 50000 nM T98711 C4UY7R 23636019 IC50 > 50000 nM T98711 CHTN58 23636020 IC50 > 50000 nM T98711 CPV52Y 23636021 IC50 > 50000 nM T98711 CD71KA 23636022 IC50 > 50000 nM T98711 C6QA3I 23636023 IC50 > 50000 nM T98711 CQ4U9X 23636024 IC50 > 50000 nM T98711 C93CLQ 23644605 IC50 = 3.8 nM T98711 CMH24N 23644647 IC50 = 5.55 nM T98711 CQ49JO 23644649 IC50 = 4.74 nM T98711 C4HV8T 23644653 IC50 = 7.8 nM T98711 C01OPD 23644658 IC50 = 4 nM T98711 CSQ9L7 23644774 IC50 = 328 nM T98711 C3AS4O 23644775 IC50 = 165 nM T98711 C2V8TA 23644776 IC50 = 45 nM T98711 C5W0NY 23644777 IC50 = 312 nM T98711 C8YQA2 23644778 IC50 = 93 nM T98711 CPO4L8 23644779 IC50 = 59 nM T98711 CSU1T2 23644780 IC50 = 23 nM T98711 C38QZE 23644781 IC50 = 3.3 nM T98711 CZH24F 23644782 IC50 = 2.6 nM T98711 CM39BI 23645223 IC50 = 1.48 nM T98711 CW8F0V 23645224 IC50 = 2580 nM T98711 CTW9J8 23645267 IC50 = 7.69 nM T98711 CRB3O6 23645269 IC50 = 6.7 nM T98711 CB8H9A 23645271 IC50 = 14 nM T98711 C34ZIH 23645273 IC50 = 7.38 nM T98711 CK2NJ4 23645289 IC50 = 1560 nM T98711 C3RP5S 23648183 IC50 = 7407 nM T98711 CQ9VY0 23648184 IC50 > 10000 nM T98711 CC0S5M 23653045 IC50 = 6401 nM T98711 CG61EZ 23765385 IC50 = 15200 nM T98711 CR8CW5 24202660 IC50 > 50000 nM T98711 CANS31 24749809 IC50 = 11.3 nM T98711 C4Z2EB 24749810 IC50 = 35.1 nM T98711 C4FVB7 24749811 IC50 = 5.44 nM T98711 CO9D4U 24799948 IC50 = 5.5 nM T98711 C6LV5R 24799949 IC50 = 36.5 nM T98711 C8JPO2 24800125 IC50 = 28 nM T98711 C64FMN 24800126 IC50 = 5.2 nM T98711 C8GKX5 24800127 IC50 = 21.7 nM T98711 C6DSC8 24800128 IC50 = 9.9 nM T98711 CW7LB1 24800129 IC50 = 15.3 nM T98711 CZ14LB 24800130 IC50 = 13.5 nM T98711 C59BPF 24800294 IC50 = 12.1 nM T98711 C07CZO 24800295 IC50 = 15.1 nM T98711 C5H3EC 24800296 IC50 = 5.5 nM T98711 C0QLV7 24800297 IC50 = 13.8 nM T98711 CAO8P0 24800298 IC50 = 10.8 nM T98711 CARE83 24800299 IC50 = 41 nM T98711 CZ0GN5 24800469 IC50 = 7.3 nM T98711 CQNB75 24825630 Ki > 100000 nM T98711 CF6W3Z 24833568 IC50 = 6820 nM T98711 C82UXG 24841476 Ki = 2450 nM T98711 C08HVP 24841478 Ki = 2400 nM T98711 CY21RE 24841480 Ki = 650 nM T98711 CVZ3G8 24845717 IC50 = 4 nM T98711 CMF3P2 24845873 IC50 = 34000 nM T98711 CR6M2L 24863097 Ki = 0.819 nM T98711 CBP1Y5 24865177 IC50 = 280 nM T98711 COR9K5 24865178 IC50 = 1830 nM T98711 CIY6F4 24865179 IC50 = 38100 nM T98711 CKB7T5 24865359 IC50 = 40900 nM T98711 CS1VB7 24865360 IC50 = 1820 nM T98711 C50JUL 24865361 IC50 = 21700 nM T98711 CH0WZ8 24865362 IC50 = 89100 nM T98711 C9W8TE 24865363 IC50 = 74100 nM T98711 C2CX0D 24879253 Ki = 0.779 nM T98711 CO3D6F 24879256 Ki = 1.187 nM T98711 CE7RA8 24879313 Ki = 0.924 nM T98711 COVB34 24879315 Ki = 13.86 nM T98711 CX60OH 24879317 Ki = 0.27 nM T98711 CW49DK 24879319 Ki = 0.725 nM T98711 C3DGL7 24879377 Ki = 0.435 nM T98711 CQM5Y4 24879379 Ki = 4.191 nM T98711 CA6WB0 24879381 Ki = 3.223 nM T98711 CRWB78 24879383 Ki = 1.872 nM T98711 C3GTP2 24879451 Ki = 5.04 nM T98711 CDI31X 24879453 Ki = 7.29 nM T98711 C51PQF 24881876 IC50 = 12.3 nM T98711 CLM2P5 24881945 IC50 = 8.06 nM T98711 CDI95B 24881949 IC50 = 7.25 nM T98711 CM5NY1 24905533 Ki = 260000 nM T98711 CBM4Q0 24905591 Ki = 3200 nM T98711 C6ZWN0 24905654 Ki = 1910 nM T98711 CW81VH 24905655 Ki = 120 nM T98711 CABV24 24936088 Ki = 19500 nM T98711 CO1ID8 24949376 IC50 = 296 nM T98711 C5VL9C 24949523 IC50 = 211 nM T98711 C2UZ4A 24949524 IC50 = 189 nM T98711 C3OV2G 24949525 IC50 = 137 nM T98711 CDY49T 25016412 IC50 = 4000 nM T98711 CVQY09 25016666 IC50 = 800 nM T98711 C2OD8R 25022724 IC50 = 4650 nM T98711 CAVC47 25033601 IC50 = 400 nM T98711 CML5I0 25053470 IC50 = 49980 nM T98711 CEM9A4 25053473 IC50 = 5890 nM T98711 CCR8V4 25053476 IC50 = 1720 nM T98711 C5XJH0 25053537 IC50 = 4590 nM T98711 C9WL5U 25053538 IC50 = 7540 nM T98711 C18HXS 25129144 IC50 = 28 nM T98711 CP91JC 25129145 IC50 = 32 nM T98711 CA2P7V 25129146 IC50 = 12 nM T98711 CD5Z2O 25129487 IC50 = 137 nM T98711 CHN93D 25145301 IC50 = 14400 nM T98711 C3P4KA 25149263 IC50 = 2090 nM T98711 CX50VY 25149264 IC50 = 293 nM T98711 CU45TK 25149265 IC50 = 1910 nM T98711 CU7EV3 25149453 IC50 = 10700 nM T98711 CB9Q1Y 25149538 IC50 = 1040 nM T98711 CEF4M1 25150256 IC50 = 30800 nM T98711 CES10Z 25150257 IC50 = 25300 nM T98711 CW5Y9S 25150356 IC50 = 10300 nM T98711 C6KSF0 25150451 IC50 = 95.8 nM T98711 CEL09B 25150452 IC50 = 876 nM T98711 CKW2Z0 25150453 IC50 = 3000 nM T98711 CB7K2G 25150454 IC50 = 416 nM T98711 CSLH31 25204947 IC50 = 334 nM T98711 C9NG2M 25205011 IC50 = 7322 nM T98711 C0TWB6 25211256 IC50 = 10000 nM T98711 CRKA79 25221268 IC50 = 116000 nM T98711 C6R3VH 25396473 Ki = 2.71 nM T98711 CKJZ59 25396479 Ki = 27.05 nM T98711 C2WPI3 27666802 IC50 = 1320 nM T98711 CL89DY 35793912 IC50 = 15300 nM T98711 CKJ82C 38864639 IC50 > 100000 nM T98711 CH4UY3 41474021 IC50 > 100000 nM T98711 CZ6KB8 41527552 IC50 = 3930 nM T98711 CJ06DE 42597801 IC50 = 60700 nM T98711 CJX2O8 42598036 IC50 = 88800 nM T98711 CX4H1M 42598039 IC50 > 100000 nM T98711 C7GO1F 42598040 IC50 = 16200 nM T98711 CE6Y3Z 42598041 IC50 = 125000 nM T98711 C0X7NH 42598042 IC50 = 71500 nM T98711 CNGR23 42598273 IC50 = 172000 nM T98711 C8K3WA 42598274 IC50 = 44000 nM T98711 CF75TP 42598275 IC50 > 100000 nM T98711 CXZ19Y 42598510 IC50 = 33200 nM T98711 CBOI16 42598737 IC50 > 10000 nM T98711 C5ROV0 42603833 IC50 = 1290 nM T98711 C2UN9H 42618134 IC50 > 100000 nM T98711 CH6X2V 42618135 IC50 > 100000 nM T98711 CCAU57 42618136 IC50 > 100000 nM T98711 C0EO3S 42618137 IC50 > 100000 nM T98711 CH21YS 42618138 IC50 > 100000 nM T98711 C2D4GJ 42637909 IC50 > 100000 nM T98711 CE4Q1Z 42637910 IC50 = 11000 nM T98711 C1E5GI 43824597 IC50 > 30000 nM T98711 C7YR8O 44224102 IC50 = 223 nM T98711 CMQ73T 44241603 IC50 = 3640 nM T98711 CNME62 44247959 IC50 = 290 nM T98711 CN80WP 44269395 IC50 = 4270 nM T98711 C2CZM3 44287477 IC50 = 910 nM T98711 CRL89F 44288141 IC50 = 920 nM T98711 C0QZG6 44288635 IC50 = 31 nM T98711 CZ9CM8 44289029 IC50 = 27 nM T98711 CWI3J4 44298002 IC50 = 1790 nM T98711 C5IS3D 44314031 IC50 = 11000 nM T98711 C4PH1U 44316259 IC50 = 216000 nM T98711 C9Y8WR 44316260 IC50 = 790000 nM T98711 C4GXD1 44316606 IC50 = 960000 nM T98711 CO6FT7 44328449 IC50 = 28000 nM T98711 C8KHN0 44328476 IC50 = 350 nM T98711 CIL4P7 44328516 IC50 = 3300 nM T98711 CK2UH8 44328517 IC50 = 2000 nM T98711 CLDZ15 44328518 IC50 = 48000 nM T98711 CD7VA3 44328527 IC50 > 50000 nM T98711 CY76FG 44328582 IC50 = 22000 nM T98711 CLB58A 44328594 IC50 > 50000 nM T98711 CY17DP 44328595 IC50 > 50000 nM T98711 CAEI14 44328600 IC50 = 2800 nM T98711 CJ10IH 44328655 IC50 = 4400 nM T98711 C27RNL 44328656 IC50 = 8800 nM T98711 CO75SD 44328657 IC50 = 2700 nM T98711 CU0VD3 44328667 IC50 = 3400 nM T98711 CYH27G 44328671 IC50 = 1000 nM T98711 CT0V8E 44328705 IC50 = 5600 nM T98711 C3T7KM 44328731 IC50 = 4400 nM T98711 CH5T7O 44328735 IC50 > 50000 nM T98711 CQ91KO 44328757 IC50 = 40000 nM T98711 C0BVX1 44328784 IC50 = 1200 nM T98711 CB9D2W 44328828 IC50 = 13000 nM T98711 CNU4R7 44328837 IC50 = 3900 nM T98711 CR97EP 44328842 IC50 = 250 nM T98711 CPE7B1 44328853 IC50 > 50000 nM T98711 CJ8Y0L 44328854 IC50 = 410 nM T98711 CR43YN 44338975 IC50 = 115 nM T98711 CUVK87 44339289 IC50 = 512 nM T98711 CT72FC 44339352 IC50 = 449 nM T98711 C0XI2G 44344490 IC50 = 88000 nM T98711 CZM80K 44344737 IC50 = 10300 nM T98711 CT1Q3S 44347198 IC50 = 50 nM T98711 CPXK27 44347214 IC50 = 2900 nM T98711 CNY9B1 44347584 IC50 = 1560 nM T98711 CVL5Y1 44347602 IC50 = 1950 nM T98711 CXD43V 44358068 IC50 = 2100 nM T98711 C05RBY 44358110 Ki = 1600 nM T98711 C3OPV1 44358179 Ki = 7500 nM T98711 CC79ZF 44361495 IC50 = 963 nM T98711 CK6QX1 44361516 IC50 = 331 nM T98711 CGHX23 44361622 IC50 = 32.6 nM T98711 C3OHM0 44361641 IC50 = 194 nM T98711 CF4GR3 44361719 IC50 = 1210 nM T98711 C0SZQ9 44362025 IC50 = 148 nM T98711 CF3H1M 44362158 IC50 = 63 nM T98711 C4L1OJ 44364861 Ki = 3250 nM T98711 CJKS01 44364863 Ki = 8600 nM T98711 CB6S7Y 44364908 IC50 = 2300 nM T98711 C39BIX 44385143 IC50 = 870.96 nM T98711 C3YO4B 44385678 IC50 = 270 nM T98711 C7Y0RT 44385890 IC50 > 2000 nM T98711 CP5FZ7 44386430 IC50 = 1410 nM T98711 CO6E7R 44386491 IC50 > 2000 nM T98711 CA5MZ0 44386492 IC50 > 2000 nM T98711 C5LXT8 44386641 IC50 > 2000 nM T98711 C61PJT 44386933 IC50 = 350 nM T98711 C9V2XH 44387832 IC50 = 3.9 nM T98711 C57WPN 44388351 IC50 = 17 nM T98711 CW09ZP 44391786 IC50 > 200000 nM T98711 CPZ3Y1 44391798 IC50 > 200000 nM T98711 C8XH3P 44391811 IC50 > 200000 nM T98711 C46ESP 44391828 IC50 > 200000 nM T98711 C56SXM 44391858 IC50 > 500000 nM T98711 CNBR80 44398165 IC50 = 24.5 nM T98711 C5P4KS 44398279 IC50 = 1.26 nM T98711 CX01VE 44398294 IC50 = 44.41 nM T98711 CN6PS1 44398377 IC50 = 10.5 nM T98711 C1M3ZD 44398397 IC50 = 209 nM T98711 C2B5HS 44398438 IC50 = 30.3 nM T98711 C7IRF1 44398566 IC50 = 74800 nM T98711 CMF05N 44409456 IC50 = 2 nM T98711 CJ35GS 44409574 IC50 = 4 nM T98711 C9ZHL5 44412131 Ki = 20.8 nM T98711 CQ12BX 44412132 Ki = 30.8 nM T98711 CHO3A1 44412135 Ki = 19.5 nM T98711 C4KN6X 44412186 IC50 = 15.8 nM T98711 CF0XV9 44417532 IC50 = 3980 nM T98711 C5MBE6 44417537 IC50 = 8490 nM T98711 C98SME 44417548 IC50 > 10000 nM T98711 CV7XP1 44417560 IC50 = 601 nM T98711 CVSZ87 44417568 IC50 > 10000 nM T98711 C0SR2L 44417569 IC50 = 9220 nM T98711 C0JYP1 44418744 IC50 = 1.38 nM T98711 CG41JA 44419699 IC50 > 10000 nM T98711 CY8RQ9 44419966 IC50 > 10000 nM T98711 CXZ52T 44419971 IC50 > 10000 nM T98711 CBD4I8 44421020 IC50 = 2300 nM T98711 C7SN0Z 44421297 IC50 = 11748.98 nM T98711 C9I7EY 44421298 IC50 = 2238.72 nM T98711 CD3SJ4 44421300 IC50 = 6456.54 nM T98711 CJ47UB 44421301 IC50 = 3630.78 nM T98711 C8GY2A 44421302 IC50 = 3388.44 nM T98711 CC64OM 44421303 IC50 = 1862.09 nM T98711 CV7RQ4 44421304 IC50 = 1819.7 nM T98711 CQ8V9A 44421305 IC50 = 1698.24 nM T98711 C6MFY8 44421520 IC50 = 136 nM T98711 CB9AO4 44421521 IC50 = 60 nM T98711 C03AEP 44421525 IC50 = 59 nM T98711 CM6IW2 44421529 IC50 = 9.6 nM T98711 CKNV25 44421531 IC50 = 54 nM T98711 CV46OY 44421933 IC50 = 63800 nM T98711 CHQ74U 44421934 IC50 = 127000 nM T98711 CM2PQ9 44421939 IC50 = 29500 nM T98711 CPM30V 44421940 IC50 = 14000 nM T98711 CX7T8G 44421945 IC50 = 2010 nM T98711 CGN9K0 44421946 IC50 = 1270 nM T98711 CR4K2Y 44421950 IC50 = 1000 nM T98711 CF0SC4 44421951 IC50 = 320 nM T98711 CH9WV0 44421967 IC50 = 46100 nM T98711 CQ6ZY2 44421972 IC50 = 3080 nM T98711 C4AF3S 44421973 IC50 = 1910 nM T98711 CO97PS 44421976 IC50 = 930 nM T98711 C1SK6X 44421982 IC50 = 1850 nM T98711 C9FZP5 44421986 IC50 = 2110 nM T98711 CTD13B 44421991 IC50 = 269000 nM T98711 CCB15K 44423472 IC50 = 29000 nM T98711 CEQ6U7 44423479 IC50 = 100 nM T98711 CO9LC6 44427467 IC50 = 279000 nM T98711 CM6GB7 44427468 IC50 > 0.00001 nM T98711 CEVO25 44427469 IC50 = 570000 nM T98711 CJ64GU 44427470 IC50 = 136000 nM T98711 CZ83QC 44427471 IC50 = 1300000 nM T98711 CPM03B 44427472 IC50 > 0.00001 nM T98711 CCJH84 44427473 IC50 > 0.00001 nM T98711 CN5CJ2 44427474 IC50 > 0.00001 nM T98711 CHQ62N 44427475 IC50 > 0.00001 nM T98711 C6WDH3 44427476 IC50 > 0.00001 nM T98711 CZTU76 44427477 IC50 > 0.00001 nM T98711 CO1NJ5 44427478 IC50 = 52900 nM T98711 CQ5G6X 44427479 IC50 > 0.00001 nM T98711 C4M7RQ 44427480 IC50 > 0.00001 nM T98711 CLS78U 44427481 IC50 = 35100 nM T98711 C5O1RW 44427482 IC50 > 0.00001 nM T98711 C0AM6W 44427483 IC50 > 0.00001 nM T98711 CE09QX 44427485 IC50 > 0.00001 nM T98711 CFMN40 44427486 IC50 > 0.00001 nM T98711 CS3AX5 44427487 IC50 > 0.00001 nM T98711 C9XM2E 44427488 IC50 > 0.00001 nM T98711 C0WMB1 44427489 IC50 > 0.00001 nM T98711 CPM76T 44427490 IC50 > 0.00001 nM T98711 CQ87RG 44427491 IC50 = 88900 nM T98711 CT38CX 44427492 IC50 > 0.00001 nM T98711 CSO3M0 44427493 IC50 = 43800 nM T98711 CDE8A1 44428745 IC50 = 10471.29 nM T98711 C0C2DX 44428836 Ki > 100000 nM T98711 CZS9U1 44428842 Ki > 100000 nM T98711 CWR3Y1 44428843 Ki > 100000 nM T98711 CUT0H7 44428844 Ki > 100000 nM T98711 C0NHI2 44435121 IC50 > 50000 nM T98711 CZ3RM2 44435219 Ki = 28 nM T98711 CIW9A7 44435348 IC50 > 1000 nM T98711 CV5Q1B 44435447 IC50 > 10000 nM T98711 CG7QK6 44435498 IC50 > 10000 nM T98711 CKP0Q3 44435526 IC50 = 1440 nM T98711 C83BXH 44435798 Ki > 100000 nM T98711 CF9SH8 44446101 Ki = 20400 nM T98711 C5K6XG 44446102 Ki = 754200 nM T98711 C7IH4Y 44446104 Ki = 161300 nM T98711 CE7M5J 44446106 Ki = 273800 nM T98711 CIQ4O9 44446113 Ki = 174500 nM T98711 CJ41TE 44550606 IC50 = 3000 nM T98711 CTYA64 44550607 IC50 = 730 nM T98711 CP0O8Q 44550608 IC50 = 70 nM T98711 CPWV46 44550725 IC50 = 1750 nM T98711 CQV8G2 44550726 IC50 = 1800 nM T98711 CNP4T9 44550727 IC50 = 850 nM T98711 CPT1O4 44550728 IC50 = 330 nM T98711 CLFZ14 44550729 IC50 = 830 nM T98711 CLVX32 44550849 IC50 = 350 nM T98711 CG1NK0 44562321 IC50 = 10000 nM T98711 CRA0U2 44562335 IC50 = 22060 nM T98711 CVA67X 44568347 Ki = 740 nM T98711 C0G8AC 44568806 IC50 = 2800 nM T98711 CJDG06 44568807 IC50 = 73 nM T98711 C0G3SJ 44580530 Ki = 1198 nM T98711 C1AO5C 44580576 Ki = 252 nM T98711 C9G1VW 44580577 Ki = 580 nM T98711 C5G2VP 44580578 Ki = 708 nM T98711 CP4FT6 44580579 Ki = 251 nM T98711 C6PLC4 44580639 Ki = 1764 nM T98711 CB1ZL8 44580640 Ki = 443 nM T98711 CQ6U4X 44580641 Ki = 173 nM T98711 CL73ZJ 44580642 Ki = 1.87 nM T98711 CK4M5S 44580643 Ki = 1.33 nM T98711 C8N4ZQ 44580644 Ki = 12.63 nM T98711 CMR90Y 44580645 Ki = 25.15 nM T98711 CWHP70 44580646 Ki = 1.77 nM T98711 CGJ3O4 44586009 IC50 = 196 nM T98711 CRJC18 44587246 IC50 = 1600 nM T98711 CM27UT 44587247 IC50 = 600 nM T98711 CKZJ17 44587345 IC50 = 29400 nM T98711 CP4G7M 44587346 IC50 = 76600 nM T98711 C37PVZ 44587494 IC50 = 4700 nM T98711 CMP67W 44587524 IC50 = 75200 nM T98711 C2CV9M 44587525 IC50 = 34400 nM T98711 CGK71P 44587544 IC50 = 3970 nM T98711 CI2L4T 44587564 IC50 = 19700 nM T98711 CIF0E9 44587921 IC50 = 142100 nM T98711 C7MW1Z 44589810 IC50 = 36800 nM T98711 CL1PQ6 44604353 IC50 > 30000 nM T98711 C34RFE 44604423 IC50 > 30000 nM T98711 C6K8GE 45049498 IC50 = 40000 nM T98711 CTBO39 45130737 IC50 = 345000 nM T98711 COF81U 45164786 IC50 = 2150 nM T98711 C5U6GX 45214445 IC50 = 21 nM T98711 CJP71Z 45261769 IC50 = 22.1 nM T98711 C2MN6D 45261778 IC50 = 24.5 nM T98711 CTYU71 45261781 IC50 = 31.6 nM T98711 CY6GX3 45261793 IC50 = 529 nM T98711 CZ16LQ 45261805 IC50 = 205 nM T98711 C67KQI 45261809 IC50 = 48.3 nM T98711 CW09OL 45261830 IC50 = 16.5 nM T98711 CY17RU 45263524 IC50 = 11600 nM T98711 CGE36P 45265144 IC50 = 34.1 nM T98711 CH6SJ9 45265175 IC50 = 25.2 nM T98711 CHA28P 45265179 IC50 = 24.8 nM T98711 COW2D8 45266157 IC50 = 660 nM T98711 CHE19F 45266158 IC50 > 10000 nM T98711 CNJ5W8 45266159 IC50 > 10000 nM T98711 C1LOR7 45266221 IC50 = 1700 nM T98711 CO9LU8 45266222 IC50 = 5200 nM T98711 CT01NJ 45267086 IC50 = 21100 nM T98711 CP5BH2 45269663 IC50 = 98100 nM T98711 C4HD1L 45269664 IC50 = 25000 nM T98711 CO4K0N 45269909 IC50 > 10000 nM T98711 CG92KC 45270503 IC50 = 175800 nM T98711 C3GF6X 45481996 IC50 = 2350 nM T98711 CQ4XH0 45481997 IC50 = 824 nM T98711 CJW20I 45482019 IC50 = 342 nM T98711 CAM26F 45482095 IC50 = 148000 nM T98711 C34LEX 45482096 IC50 = 31000 nM T98711 CK4Z8S 45482098 IC50 = 50000 nM T98711 C2CNM7 45482099 IC50 = 16100 nM T98711 CHMS72 45482100 IC50 = 133000 nM T98711 CYSP25 45482101 IC50 = 4200 nM T98711 CPT8J4 45482102 IC50 = 13400 nM T98711 C8ETA6 45482104 IC50 = 760 nM T98711 CDPT02 45482105 IC50 = 22000 nM T98711 CRO52I 45482106 IC50 = 140 nM T98711 CKE2N4 45487235 IC50 = 117 nM T98711 CG5W3E 45487242 IC50 = 0.15 nM T98711 C2VC7M 45487244 IC50 = 16 nM T98711 CF8M9K 45487246 IC50 = 323 nM T98711 CBTU95 45487247 IC50 = 18 nM T98711 C6B1IN 45487248 IC50 = 27 nM T98711 CG1ZJ8 45487252 IC50 = 86 nM T98711 CSQ78Z 45487253 IC50 = 297 nM T98711 C2SH7T 45487255 IC50 = 39 nM T98711 CLS2D9 45487263 IC50 = 32 nM T98711 CMJB89 45487264 IC50 = 9.6 nM T98711 CJ20LD 45487265 IC50 = 6.4 nM T98711 CBHD59 45487269 IC50 = 2609 nM T98711 C7S8KN 45487275 IC50 = 1057 nM T98711 CQFC83 45488333 IC50 > 5000 nM T98711 CW68OR 45490978 IC50 = 9570 nM T98711 C5IOS9 45490990 IC50 = 37400 nM T98711 C91TIQ 46204460 IC50 = 450300 nM T98711 CIG1O6 46211767 IC50 = 16210 nM T98711 CC64KH 46227076 IC50 = 19 nM T98711 C1MSE9 46228657 IC50 = 144000 nM T98711 C31MLQ 46228658 IC50 = 21100 nM T98711 CT9CI3 46228685 IC50 = 7930 nM T98711 CIK7S8 46228686 IC50 = 98100 nM T98711 C2V4QP 46228687 IC50 = 29900 nM T98711 CC85MY 46228688 IC50 = 22500 nM T98711 CE86KJ 46228721 IC50 = 11400 nM T98711 C7CY5S 46228722 IC50 = 22900 nM T98711 C7W8OG 46228723 IC50 = 11900 nM T98711 CK62AH 46228724 IC50 = 11900 nM T98711 C20GZR 46228760 IC50 = 3520 nM T98711 C4O9CE 46228761 IC50 = 99800 nM T98711 CLUW07 46228762 IC50 = 10000 nM T98711 CJ5YZ9 46228787 IC50 = 2700 nM T98711 CJ2D5H 46228788 IC50 = 7700 nM T98711 CJG67U 46228789 IC50 = 20500 nM T98711 CTBX50 46228809 IC50 = 33000 nM T98711 C6O3FS 46228810 IC50 = 90300 nM T98711 C0PHL3 46228811 IC50 = 135000 nM T98711 C9IE5S 46228812 IC50 = 72800 nM T98711 C7POL5 46228839 IC50 = 8050 nM T98711 C1E3LQ 46228840 IC50 = 5010 nM T98711 CEBO01 46229144 Ki = 9 nM T98711 CEL2V1 46229162 Ki = 250 nM T98711 C7Q6RX 46231880 IC50 = 5000 nM T98711 CH4K6D 46232763 IC50 = 10250 nM T98711 CH9EG0 46232810 IC50 = 4800 nM T98711 CI3DT1 46232813 IC50 = 52 nM T98711 C6C1ER 46232814 IC50 = 201 nM T98711 C0VIS5 46854881 IC50 = 20 nM T98711 CD0Q4G 46855034 IC50 = 6.5 nM T98711 CBO8D7 46863225 IC50 = 7900 nM T98711 CJ16FO 46866088 IC50 = 800 nM T98711 CG0UA1 46877971 IC50 = 1300 nM T98711 CX7J9D 46880263 IC50 = 2360000 nM T98711 CM6PJ3 46880264 IC50 = 1270000 nM T98711 C61VGD 46880266 IC50 = 1380000 nM T98711 C5G4FV 46880955 IC50 = 78000 nM T98711 CHNP43 46888221 IC50 > 200000 nM T98711 CZQL62 46897981 IC50 = 210 nM T98711 C4TWY7 46897983 IC50 = 140 nM T98711 CDG49K 46897985 IC50 = 43 nM T98711 CA7CK3 46897987 IC50 = 51 nM T98711 CY7ZW5 46937311 IC50 = 0.86 nM T98711 CXJ04C 49796971 IC50 = 406 nM T98711 CC86IT 49799305 IC50 = 130 nM T98711 CZYU91 49801688 IC50 = 4480 nM T98711 C35VYE 49845186 IC50 = 2450000 nM T98711 C4FHO0 49845187 IC50 = 1620000 nM T98711 CA9E5S 49845368 IC50 = 2140000 nM T98711 C6SE1Z 49845372 IC50 = 430000 nM T98711 C6BC2U 49845373 IC50 = 1580000 nM T98711 C7IJ3C 49857726 Ki > 100000 nM T98711 C04NYX 49857906 Ki > 100000 nM T98711 CDT4Y6 49857907 Ki > 100000 nM T98711 C5XS3G 49857908 Ki > 100000 nM T98711 CHRB62 49857909 Ki > 100000 nM T98711 CV7J6X 49857910 Ki > 100000 nM T98711 CYU39N 49857911 Ki > 100000 nM T98711 C5WZL0 49857912 Ki > 100000 nM T98711 CCG80U 49858100 Ki > 100000 nM T98711 CCN05H 49858101 Ki > 100000 nM T98711 C2OK0N 50874404 IC50 > 50000 nM T98711 CJE91N 50874405 IC50 > 50000 nM T98711 CTQX80 50942800 IC50 = 60 nM T98711 C8DS0J 50942802 IC50 = 16 nM T98711 CA43KF 51026481 IC50 = 170 nM T98711 C9VXK3 51039357 IC50 = 64000 nM T98711 CU36CR 51039359 IC50 = 25000 nM T98711 C8X5WJ 51039361 IC50 = 600 nM T98711 C1BA7H 51039363 IC50 = 1000 nM T98711 C4RQZ0 51039365 IC50 = 4000 nM T98711 C61UMV 51042596 IC50 = 154000 nM T98711 C2I3RA 51346780 IC50 = 1600 nM T98711 C4MH6G 51346832 IC50 = 400 nM T98711 C9AZ3J 51357040 IC50 > 10000 nM T98711 C8T1BE 51357043 IC50 > 10000 nM T98711 C3BRM2 51357044 IC50 > 10000 nM T98711 CIZ96K 51357316 IC50 > 10000 nM T98711 C5RXF2 51357319 IC50 > 10000 nM T98711 C6G9SM 51357595 Ki = 2100 nM T98711 C1R0DP 51357597 Ki = 79 nM T98711 CU0I5S 51357598 Ki = 2600 nM T98711 CE3H6X 51357599 Ki = 380 nM T98711 CGV79B 51357600 IC50 > 10000 nM T98711 C6S1KB 51357868 IC50 > 10000 nM T98711 C7QPU6 52110752 IC50 = 22000 nM T98711 CD52WQ 52111959 IC50 = 11400 nM T98711 C0LG4K 52899556 IC50 = 58600 nM T98711 CEGS83 52940502 IC50 = 940 nM T98711 C5PJL4 52940842 IC50 = 97000 nM T98711 C3F7VC 52946604 IC50 = 230 nM T98711 CQRK41 52948055 IC50 = 64000 nM T98711 C3ORW4 52949034 IC50 = 920 nM T98711 C8ZKR5 52952236 IC50 = 36 nM T98711 C4JG6W 52952244 IC50 = 620 nM T98711 CIO3V4 52952919 IC50 = 35000 nM T98711 C61YEU 52952920 IC50 = 11000 nM T98711 C9T8YE 52952921 IC50 = 9700 nM T98711 CDYC75 52952922 IC50 = 21900 nM T98711 C4Z6WM 52952958 IC50 = 39000 nM T98711 C8XV3H 52993127 IC50 = 9010 nM T98711 CPMW48 53231243 IC50 = 209000 nM T98711 CD4NP3 53231341 IC50 = 144000 nM T98711 C6RE1G 53231342 IC50 = 145000 nM T98711 CK64RX 53231343 IC50 = 179000 nM T98711 C4VE2O 53231344 IC50 = 68000 nM T98711 CNC2D0 53231345 IC50 = 21000 nM T98711 C0Z3AM 53231442 IC50 = 34000 nM T98711 C5A3YX 53231443 IC50 = 10400 nM T98711 CPM56F 53231444 IC50 = 23000 nM T98711 CO40KS 53231445 IC50 = 24200 nM T98711 C5M0OA 53242257 Ki = 1740 nM T98711 C9EL0U 53306553 IC50 = 3326 nM T98711 C3DS7L 53316786 IC50 = 241000 nM T98711 C67YGU 53320725 IC50 = 150 nM T98711 CY9HE5 53320727 IC50 = 110 nM T98711 CF0AC4 53320729 IC50 = 19000 nM T98711 CY7J8V 53320731 IC50 = 1300 nM T98711 CXB5G7 53321044 IC50 > 10000 nM T98711 C0DUN8 53321516 IC50 = 3000 nM T98711 CFKJ51 53322024 Ki = 100 nM T98711 CH1O9A 53322846 IC50 = 700 nM T98711 C26USF 53323382 IC50 = 700 nM T98711 CZT5X1 53323384 IC50 = 2400 nM T98711 C2RJQ1 53324171 IC50 = 2600000 nM T98711 CE0W5F 53324336 IC50 = 1900 nM T98711 CM1KA7 53324700 IC50 = 5100 nM T98711 C1XL0O 53324702 IC50 = 4400 nM T98711 C4YWN2 53326005 IC50 = 600 nM T98711 CW8ZV1 53326729 IC50 = 2000 nM T98711 CK45JD 53361165 IC50 = 0.0449 nM T98711 CTSC36 53361167 IC50 = 0.0354 nM T98711 CIP6E3 53361169 IC50 = 0.0212 nM T98711 CWK2J9 54097201 IC50 = 8130 nM T98711 CDCR53 54577393 IC50 = 24.8 nM T98711 CUSF85 54577394 IC50 = 63.7 nM T98711 CVJA50 54577395 IC50 = 1660 nM T98711 CXOH83 54577607 IC50 = 28.6 nM T98711 CD8PN5 54580372 IC50 = 871000 nM T98711 CT2L8P 54580374 IC50 = 308000 nM T98711 C7DH8A 54580376 IC50 = 200 nM T98711 C1IE9P 54580388 IC50 = 501 nM T98711 C3ENI1 54580389 IC50 > 10000 nM T98711 CN20LZ 54581356 IC50 > 10000 nM T98711 C6KVB5 54581375 IC50 = 700 nM T98711 CBH4L1 54581388 IC50 > 1000 nM T98711 C23NPW 54582394 IC50 = 13000 nM T98711 CH60OU 54582403 IC50 > 10000 nM T98711 C1MZ0J 54582404 IC50 > 10000 nM T98711 CX8N5Y 54582406 IC50 > 10000 nM T98711 CXVQ08 54583385 IC50 = 1430 nM T98711 C7WS9L 54583386 IC50 = 333 nM T98711 C8NXY5 54583387 IC50 = 679 nM T98711 C21PHC 54584309 IC50 = 224 nM T98711 CZ8E5U 54584310 IC50 = 217 nM T98711 CH7JX8 54584326 IC50 = 20000 nM T98711 CZW86O 54584337 IC50 > 10000 nM T98711 CVB76W 54584338 IC50 = 554 nM T98711 CW8EU4 54585277 IC50 > 10000 nM T98711 C9VCF6 54585278 IC50 > 10000 nM T98711 C9ZSE5 54585303 IC50 = 32000 nM T98711 C2SQ7Y 54586227 IC50 = 5375 nM T98711 CNEB14 54586228 IC50 = 1343 nM T98711 C97ESH 54586244 IC50 = 400 nM T98711 CUR47F 54587253 IC50 = 477 nM T98711 CY9X6B 54587254 IC50 = 653 nM T98711 C0WMB8 54587272 IC50 = 48000 nM T98711 C8PH1A 54587274 IC50 = 800 nM T98711 CV3F8K 54587276 IC50 = 6000 nM T98711 C75HCV 54587283 IC50 > 10000 nM T98711 C9KL7N 54587284 IC50 = 2948 nM T98711 C3Y1NF 54604881 IC50 > 5000 nM T98711 C4JOA7 54753261 IC50 = 1100 nM T98711 CE1ZN5 54754513 IC50 > 200000 nM T98711 CQ1MY9 54768917 IC50 = 101 nM T98711 C61LVE 54768918 IC50 = 90.5 nM T98711 C6FD9U 54768919 IC50 = 42.8 nM T98711 CD19BL 54768920 IC50 = 38.1 nM T98711 CVQ80D 54768921 IC50 = 14.7 nM T98711 CSUP59 54768922 IC50 = 101 nM T98711 CAP3I8 54769156 IC50 = 7280 nM T98711 C9O1JY 54769157 IC50 = 41.4 nM T98711 CFYX02 56649564 IC50 = 8570 nM T98711 C9TNA0 56926078 IC50 = 3160 nM T98711 CH46AD 56926079 IC50 = 3580 nM T98711 CJ31RE 56930476 IC50 = 30.6 nM T98711 CNYF34 56930477 IC50 = 205000 nM T98711 C0J2NP 56930478 IC50 = 398 nM T98711 CDQ32W 56933910 IC50 = 3780 nM T98711 CXNJ86 56933912 IC50 = 119000 nM T98711 CLB67G 56934051 IC50 = 26100 nM T98711 C4ZBA5 56934056 IC50 > 100000 nM T98711 CMA7L0 56954888 IC50 = 0.08 nM T98711 C4M1ET 56954890 IC50 = 0.038 nM T98711 C8XCI0 56954891 IC50 = 0.1 nM T98711 CHV8U3 56954986 IC50 = 0.1 nM T98711 CV3X9D 56954987 IC50 = 0.1 nM T98711 C0JCZ2 56954989 IC50 = 15 nM T98711 CTB71C 56954996 IC50 = 0.15 nM T98711 C4A6LW 56955097 IC50 = 50 nM T98711 CC7Y5O 56955099 IC50 = 1.5 nM T98711 C25KBX 56955100 IC50 = 1.5 nM T98711 C9XO0M 56955109 IC50 = 1 nM T98711 COE65B 56955111 IC50 = 0.8 nM T98711 C4U9FZ 56955198 IC50 = 5 nM T98711 C9I3AY 56955199 IC50 = 2.5 nM T98711 C2EY4O 56955292 IC50 = 30 nM T98711 C2M6DQ 56955293 IC50 = 95 nM T98711 CHA1I9 57342686 IC50 > 3000000 nM T98711 CZBE16 57342689 IC50 = 375.9 nM T98711 CC76WY 57342690 IC50 = 42.6 nM T98711 CVK98Q 57383995 IC50 = 1.57 nM T98711 CHB7N4 57390352 IC50 > 200000 nM T98711 CNM3O8 57390398 IC50 = 656000 nM T98711 CZDN40 57391125 IC50 = 78800 nM T98711 COAM20 57392136 IC50 > 200000 nM T98711 C5D7HF 57396286 IC50 = 12.1 nM T98711 CJE63A 57397445 IC50 > 200000 nM T98711 CZ3KT7 57402629 IC50 > 200000 nM T98711 CPUM70 59740711 IC50 = 2030 nM T98711 CV2G0U 60144120 IC50 = 82000 nM T98711 CVO2Z4 60148583 IC50 = 549.2 nM T98711 C4F1PE 60165327 IC50 = 6.4 nM T98711 CO58SL 60661850 IC50 > 100000 nM T98711 C4KS0V 62707049 IC50 = 11.2 nM T98711 CNW04I 62707050 IC50 = 1.71 nM T98711 C1U2FD 62707051 IC50 = 27.6 nM T98711 CZV81L 64338500 IC50 > 100000 nM T98711 CYRU28 66573467 IC50 > 10000 nM T98711 CDVT38 66573526 IC50 > 10000 nM T98711 CSA1R0 66573527 IC50 > 10000 nM T98711 CN0H5V 66573528 IC50 = 9370 nM T98711 CE52KG 66573529 IC50 > 10000 nM T98711 CMXZ21 66573530 IC50 > 10000 nM T98711 CC9Z1H 66573531 IC50 > 10000 nM T98711 C3W0YV 66573584 IC50 > 10000 nM T98711 C9QK4S 66573585 IC50 > 10000 nM T98711 C32IQA 66573586 IC50 > 10000 nM T98711 C0YE1R 68259803 IC50 = 81600 nM T98711 CJ7M5L 70683121 IC50 = 74.2 nM T98711 C09ICA 70684451 IC50 = 211 nM T98711 CD16OS 70684889 IC50 = 1500 nM T98711 CPO69B 70685195 IC50 = 44.2 nM T98711 C9HE4I 70685196 IC50 = 51.3 nM T98711 CXY5N6 70686590 IC50 = 41.2 nM T98711 CN8XT5 70687043 IC50 = 260 nM T98711 C5WOI8 70689140 IC50 = 6600 nM T98711 C7LMF4 70689416 IC50 = 24.6 nM T98711 CE4OI8 70689417 IC50 = 75.2 nM T98711 CV1DC5 70689418 IC50 = 35.1 nM T98711 CU2XC0 70690775 IC50 = 137 nM T98711 C8RPA4 70692911 IC50 = 63.7 nM T98711 CC3Y2P 70692912 IC50 = 33.7 nM T98711 CW8AX2 70692913 IC50 = 1520 nM T98711 C6AHB9 70693333 IC50 > 10000 nM T98711 CA7CP6 70693341 IC50 = 580 nM T98711 C2LV8M 70694951 IC50 = 126 nM T98711 CC39LU 70695442 IC50 = 670 nM T98711 C1U2SF 70695443 IC50 = 1700 nM T98711 CF9EO8 70697005 IC50 = 77.8 nM T98711 CWO7H5 70697453 IC50 > 10000 nM T98711 CN93VA 71330901 IC50 = 4700 nM T98711 C7AJN9 71449137 IC50 = 16.4 nM T98711 CX8KG3 71449167 IC50 > 50000 nM T98711 CRC86Q 71449660 Ki = 56 nM T98711 CVF86W 71449711 IC50 = 400 nM T98711 C06WZI 71449712 IC50 = 1970 nM T98711 C24OJQ 71451471 Ki = 97 nM T98711 CVKC68 71451473 Ki = 93 nM T98711 C7NS9H 71451521 IC50 = 3180 nM T98711 CDES68 71451522 IC50 = 23000 nM T98711 CJ1AS9 71452935 IC50 = 61.2 nM T98711 C5CK7V 71453297 Ki = 55 nM T98711 CJD10W 71453346 IC50 = 136000 nM T98711 CYVB31 71453347 IC50 = 6600 nM T98711 CTJ6W4 71453348 IC50 = 880 nM T98711 CN14WJ 71453349 IC50 = 43900 nM T98711 CJ4B5X 71453350 IC50 = 2510 nM T98711 CHGF12 71453367 IC50 = 1890 nM T98711 C28XSH 71454519 IC50 = 31.1 nM T98711 C2JYF6 71455057 IC50 = 88900 nM T98711 C4JDI7 71455058 IC50 = 2880 nM T98711 CL4F6Z 71455059 IC50 = 48 nM T98711 CAJ7O6 71456744 IC50 = 20360 nM T98711 CL02JI 71456801 Ki = 166 nM T98711 CC7F6N 71456803 Ki = 82 nM T98711 C2B8LY 71456805 Ki = 99 nM T98711 CA93KH 71456856 IC50 = 7470 nM T98711 C1D6KG 71456857 IC50 = 60100 nM T98711 CP1OY9 71456858 IC50 = 89100 nM T98711 CP4K8E 71456859 IC50 = 21000 nM T98711 C10XZB 71458090 IC50 > 50000 nM T98711 C3ZU1K 71458289 IC50 = 50.1 nM T98711 CV5TX6 71458713 IC50 = 55600 nM T98711 CH7L4U 71458714 IC50 = 81200 nM T98711 C35XHD 71458715 IC50 = 1810 nM T98711 C3ASY5 71458716 IC50 = 3010 nM T98711 C0YS7T 71460136 IC50 = 9.2 nM T98711 CXHM16 71460484 Ki = 2360 nM T98711 C2JBI7 71462190 Ki = 66 nM T98711 CTY0B6 71462239 IC50 = 3000 nM T98711 CBM3S6 71462240 IC50 = 9420 nM T98711 C5YHW6 71462241 IC50 = 1370 nM T98711 C7DQL5 71475219 IC50 = 499000 nM T98711 C8ZDA2 71492183 IC50 = 375300 nM T98711 CLN29O 71587645 Ki = 0.131 nM T98711 CD5K9Y 71602709 IC50 = 8270 nM T98711 CLGH80 71653617 IC50 = 108.97 nM T98711 CEI5B1 71653619 IC50 = 57.3 nM T98711 CC45NP 71653620 IC50 = 82.34 nM T98711 CA81JD 71653759 IC50 = 30.47 nM T98711 CW9EZ1 71653760 IC50 = 120.13 nM T98711 CIFJ03 71653761 IC50 = 92.42 nM T98711 C1LVE7 71653762 IC50 = 37.57 nM T98711 CRYS21 71653918 IC50 = 67.31 nM T98711 C25PJH 71653919 IC50 = 61.69 nM T98711 CJ9LX8 71653920 IC50 = 7.1 nM T98711 CY9Z1K 71654077 IC50 = 76.89 nM T98711 CMFG63 71654078 IC50 = 58 nM T98711 CSW15Q 71654079 IC50 = 29.28 nM T98711 COH09E 71654080 IC50 = 34.75 nM T98711 C7Q5ON 71654239 IC50 = 55.25 nM T98711 CSF8E7 71654240 IC50 = 35.98 nM T98711 CS5M3R 71654241 IC50 = 29.56 nM T98711 CT8WV6 71654242 IC50 = 12.44 nM T98711 CFMB35 71723450 IC50 > 100000 nM T98711 CV16HS 71723451 IC50 > 100000 nM T98711 C7U5ER 71723452 IC50 = 71920 nM T98711 CF2VL4 71723589 IC50 = 2260 nM T98711 COT21H 71723590 IC50 > 100000 nM T98711 C9RLM5 71769057 Ki = 16820 nM T98711 C9NYJ2 71770939 Ki = 624425 nM T98711 CN06CX 71770940 Ki = 282620 nM T98711 C4R9EZ 72374595 IC50 = 8130 nM T98711 CK38PO 72374596 IC50 > 10000 nM T98711 C0FN4W 72374597 IC50 > 10000 nM T98711 C9LNA8 72376170 IC50 = 9410 nM T98711 CULW84 72376171 IC50 = 5620 nM T98711 CY19TH 72376172 IC50 = 8390 nM T98711 C45BXP 72543919 IC50 = 22500 nM T98711 C78ZPH 72544154 IC50 = 14700 nM T98711 CKAG40 72544155 IC50 = 360 nM T98711 CPH96F 72544156 IC50 = 18700 nM T98711 CE49KY 72544381 IC50 > 20000 nM T98711 CTW28Y 72544382 IC50 = 16400 nM T98711 C6TQ7M 72545286 IC50 = 9980 nM T98711 CBL6J5 72545287 IC50 = 7770 nM T98711 CKY67A 72724835 IC50 = 1000 nM T98711 C59UPS 72724837 IC50 = 7700 nM T98711 CA16UV 72724839 IC50 = 350 nM T98711 CTB2A1 72724841 IC50 = 370 nM T98711 C02IHQ 72724843 IC50 = 700 nM T98711 CGJ2T1 72724905 IC50 = 2200 nM T98711 C5Z4BW 72724907 IC50 = 2000 nM T98711 CJA54D 72724909 IC50 = 1700 nM T98711 C3OUZ2 72724911 IC50 = 3200 nM T98711 CY2M3K 72724913 IC50 = 900 nM T98711 CPWA14 72724915 IC50 = 680 nM T98711 C1LH5Z 72725438 Ki = 0.06 nM T98711 C6CJT1 72725439 Ki = 8.26 nM T98711 C3K0SD 72725440 Ki = 40.9 nM T98711 CS1TQ7 72725488 Ki = 61.77 nM T98711 C9ZB1M 72725489 Ki = 21.26 nM T98711 C53XHE 73346133 IC50 = 470 nM T98711 C9RWV8 73352248 IC50 > 10000 nM T98711 COKX05 73352249 IC50 > 10000 nM T98711 C45GXL 73356781 IC50 > 10000 nM T98711 CGD8R4 73671789 IC50 = 2100 nM T98711 CV13PU 76310709 IC50 > 10000 nM T98711 CZ49PQ 76311731 IC50 = 26000 nM T98711 CGI2O5 76317912 IC50 > 25000 nM T98711 C1I2UO 76317913 IC50 = 970 nM T98711 CE5M1O 76317914 IC50 > 10000 nM T98711 CC1PL3 76318071 IC50 = 1370 nM T98711 C4M8ZY 76321622 IC50 > 10000 nM T98711 CSXH87 76321623 Ki = 220 nM T98711 C1W8HB 76325234 Ki = 1200 nM T98711 CO05NW 76325235 Ki = 1000 nM T98711 C5AV9G 76328789 Ki = 28 nM T98711 C4QH5I 76328790 IC50 > 10000 nM T98711 C30AMV 76328791 IC50 > 100000 nM T98711 CB1KJ6 76328792 Ki = 2900 nM T98711 CEKP26 76328944 IC50 = 2590 nM T98711 CTG51J 76336093 IC50 > 10000 nM T98711 C48RZI 76336227 IC50 = 920 nM T98711 C57UTS 77108165 IC50 = 3700 nM T98711 C0JCK7 77461631 IC50 = 7224 nM T98711 C7GX5I 78350462 IC50 = 540 nM T98711 CA3YL2 78426937 IC50 > 40000 nM T98711 CR0H5Q 78427074 IC50 > 40000 nM T98711 C2ZOJ4 78427075 IC50 = 32000 nM T98711 CJCL87 78427076 IC50 = 15900 nM T98711 CH3NJ9 78427077 IC50 > 40000 nM T98711 CR84AG 78427078 IC50 > 40000 nM T98711 CV9DO7 78427079 IC50 > 40000 nM T98711 C4US9B 78427204 IC50 = 3100 nM T98711 CS0N1V 78427205 IC50 = 18900 nM T98711 CG46NS 78427206 IC50 > 40000 nM T98711 C3WL0E 78427207 IC50 = 14600 nM T98711 CK5X0H 78427208 IC50 = 12100 nM T98711 CN6L8C 78427209 IC50 = 21300 nM T98711 CCE8Q9 78427338 IC50 = 6500 nM T98711 C0CL4Y 80772460 IC50 = 5000 nM T98711 CI5GO1 83453608 IC50 = 18000 nM T98711 C5MC7H 85470203 IC50 = 5990 nM T98711 CHXN26 85852196 Ki = 341000 nM T98711 CB3ZI5 86294786 IC50 = 5830 nM T98711 CXC80P 86581945 IC50 = 9200 nM T98711 C8CF5A 88749792 IC50 > 100000 nM T98711 CRZ0W3 90356636 IC50 = 14900 nM T98711 CI3ZW5 90356648 IC50 > 40000 nM T98711 C85UDM 90356741 IC50 > 40000 nM T98711 C2Z5FB 90356750 IC50 > 40000 nM T98711 CYB89Q 90356760 IC50 = 14100 nM T98711 CW8N4S 90356765 IC50 > 40000 nM T98711 C3NKB2 90356879 IC50 = 29200 nM T98711 CO1RJ4 90356882 IC50 = 27800 nM T98711 C9UI0O 90356903 IC50 > 40000 nM T98711 CO2HX6 90356923 IC50 = 17600 nM T98711 C52SQL 90356955 IC50 > 40000 nM T98711 C5YD7M 90356964 IC50 = 33200 nM T98711 C31XOK 90357088 IC50 > 40000 nM T98711 C0P3IL 90357101 IC50 > 40000 nM T98711 CR54TH 90357102 IC50 = 17900 nM T98711 CBJ4I2 90357105 IC50 > 40000 nM T98711 CDXO02 90357107 IC50 = 24700 nM T98711 CY9T0A 90357109 IC50 > 40000 nM T98711 CWKM49 90357121 IC50 = 21100 nM T98711 CZ7CG4 90357147 IC50 = 23400 nM T98711 C1FKL7 90357154 IC50 > 40000 nM T98711 C1LO9P 90357159 IC50 = 20100 nM T98711 CYDQ90 90357180 IC50 > 40000 nM T98711 C3I9SK 90357196 IC50 = 18400 nM T98711 CSY64P 90357367 IC50 = 4200 nM T98711 C3YJ1K 90643449 IC50 = 333300 nM T98711 CJTA92 90643450 IC50 = 362300 nM T98711 CP72GI 90643451 IC50 = 384600 nM T98711 C5SAX0 90643452 IC50 = 409000 nM T98711 CZTO98 90643453 IC50 = 430000 nM T98711 CL4Z8B 90643454 IC50 = 451000 nM T98711 C0LKB7 90643455 IC50 = 452000 nM T98711 C6RY4Q 90643456 IC50 = 454500 nM T98711 CW28SA 90643457 IC50 = 500000 nM T98711 CO3G4W 90643458 IC50 = 512000 nM T98711 CWG1P9 90643459 IC50 = 568000 nM T98711 CS0N9O 90643460 IC50 = 585000 nM T98711 CN8XQ5 90643461 IC50 = 100 nM T98711 CR67MP 90643462 IC50 = 248000 nM T98711 C0DIJ2 90643463 IC50 = 294000 nM T98711 C1E8XY 90643464 IC50 = 295000 nM T98711 CJW74Q 90643465 IC50 = 297600 nM T98711 C6Z3CW 90643468 IC50 = 19700 nM T98711 CHW4X8 90643469 IC50 = 42400 nM T98711 CU8A1S 90643470 IC50 = 43600 nM T98711 CEAB94 90643471 IC50 = 65500 nM T98711 CUO8H3 90643472 IC50 = 83300 nM T98711 CTVJ69 90645106 IC50 = 43660 nM T98711 CYW8G5 90645107 IC50 = 38530 nM T98711 C1R6LU 90645108 IC50 = 12340 nM T98711 C5U8JA 90645109 IC50 > 100000 nM T98711 C8CKM6 90645110 IC50 = 65270 nM T98711 CYN86M 90645111 IC50 = 88930 nM T98711 C3EAW0 90645112 IC50 = 14660 nM T98711 C4XF1V 90645113 IC50 > 100000 nM T98711 C30WLJ 90645114 IC50 > 100000 nM T98711 CG6YO8 90645115 IC50 > 100000 nM T98711 CJZ4X5 90645116 IC50 > 100000 nM T98711 CO20MQ 90645117 IC50 = 19740 nM T98711 C8QHF2 90645118 IC50 = 22650 nM T98711 CVPN52 90645119 IC50 > 100000 nM T98711 CXHK56 90645120 IC50 > 100000 nM T98711 CF4EB2 90645121 IC50 > 100000 nM T98711 CB2E7N 90645122 IC50 > 100000 nM T98711 CR2VS4 90645123 IC50 > 100000 nM T98711 C1ZYO3 90645124 IC50 > 100000 nM T98711 C2CI1S 90645125 IC50 > 100000 nM T98711 C40YGU 90645126 IC50 > 100000 nM T98711 C4R7BX 90645127 IC50 > 100000 nM T98711 CMN7Z9 90645128 IC50 > 100000 nM T98711 C62RBA 90645129 IC50 = 66750 nM T98711 CXU48E 90645130 IC50 = 56920 nM T98711 CYG4D2 90645131 IC50 > 100000 nM T98711 CPM6V1 90645132 IC50 > 100000 nM T98711 CP1OU8 90645133 IC50 > 100000 nM T98711 CAB7V8 90654202 IC50 = 4.28 nM T98711 CX03IG 90654705 IC50 = 3850 nM T98711 C93PIK 90654706 IC50 = 1250 nM T98711 CWLF50 90654707 IC50 = 5190 nM T98711 CP5T0F 90654708 IC50 = 7650 nM T98711 CP4U3I 90654791 IC50 = 36200 nM T98711 C62CPS 90654792 IC50 = 32100 nM T98711 CLI41J 90654793 IC50 = 39150 nM T98711 CNJ69Y 90654795 IC50 = 52760 nM T98711 CWQ16H 90654796 IC50 = 39410 nM T98711 CD1FR7 90654797 IC50 = 18010 nM T98711 CWF6X2 90654981 IC50 = 5.66 nM T98711 CMC46P 90655184 IC50 = 950 nM T98711 C12GDL 90655186 IC50 = 1070 nM T98711 C36VCM 90655188 IC50 = 1460 nM T98711 CL7PI9 90655190 IC50 = 350 nM T98711 CZ18NX 90655191 IC50 = 620 nM T98711 CH7C4F 90655192 IC50 = 265 nM T98711 CMJ31X 90655193 IC50 = 513 nM T98711 C3IZ2O 90655195 IC50 = 1100 nM T98711 CG69TU 90655196 IC50 = 645 nM T98711 C6WH0F 90655198 IC50 = 510 nM T98711 CT2N6S 90656307 IC50 = 23730 nM T98711 CTXS90 90656308 IC50 = 10590 nM T98711 CHJ71K 90656309 IC50 = 15900 nM T98711 C1FSU2 90656310 IC50 = 12900 nM T98711 CMAJ10 90656311 IC50 = 21710 nM T98711 CY0KN8 90656312 IC50 = 9290 nM T98711 CF9A7K 90656313 IC50 = 16700 nM T98711 C2I0ZP 90656314 IC50 = 3430 nM T98711 CKXS95 90656315 IC50 = 11170 nM T98711 CP4D2I 90656316 IC50 = 6020 nM T98711 CDV62L 90656317 IC50 = 6420 nM T98711 C2E0NT 90656318 IC50 = 3250 nM T98711 CS4ZQ0 90656319 IC50 = 2270 nM T98711 CNCZ35 90663111 IC50 > 50000 nM T98711 CP48CG 90663114 IC50 > 50000 nM T98711 C6JS8W 90664279 IC50 = 700 nM T98711 CY86BC 90664299 IC50 = 1931 nM T98711 C7NGZ1 90664300 IC50 = 218 nM T98711 C1KOL2 90664301 IC50 = 1076 nM T98711 C30SQY 90664402 IC50 = 331 nM T98711 CKU86A 90664403 IC50 = 1391 nM T98711 CM4NF3 90664404 IC50 = 1622 nM T98711 CKL69C 90664470 IC50 = 87.1 nM T98711 CL65ZG 90664552 IC50 = 586 nM T98711 C0GN8Y 90664609 IC50 = 43.3 nM T98711 C05QSY 90664655 Ki = 379700 nM T98711 CPE7N6 90664658 IC50 = 88.7 nM T98711 CYGT83 90664665 IC50 = 234 nM T98711 CO82LG 90664779 IC50 = 136 nM T98711 C90OVC 90664784 IC50 = 1074 nM T98711 C4EA8P 90664797 IC50 = 55 nM T98711 C7H6ZG 90664851 IC50 = 26.6 nM T98711 C3AON4 90664852 IC50 = 73.3 nM T98711 CI0NQ2 90664853 IC50 = 86.8 nM T98711 CLQ1F4 90664854 IC50 = 47.4 nM T98711 CFK51Z 90664907 IC50 = 66.3 nM T98711 CI1T4S 90664976 IC50 = 133 nM T98711 CXB25V 90664977 IC50 = 27.2 nM T98711 C1DN7L 90664978 IC50 = 76.6 nM T98711 CFPS72 90665034 Ki = 273400 nM T98711 CW36ZP 90665154 IC50 = 72.7 nM T98711 C80QZK 90665217 IC50 = 139 nM T98711 CB70OR 90667344 IC50 = 30000 nM T98711 C17ZXD 90667346 IC50 = 6700 nM T98711 C2JT9Z 90667348 IC50 = 65000 nM T98711 C8SUR1 90667350 IC50 = 10000 nM T98711 CTDR94 90667352 IC50 = 60000 nM T98711 CYIJ47 90667354 IC50 > 1000000 nM T98711 C6J7ZA 90667356 IC50 = 4200 nM T98711 CTWS98 90667358 IC50 = 1600 nM T98711 C1PY0T 90676323 IC50 = 11700 nM T98711 CQ76YM 90679728 IC50 = 34673.69 nM T98711 C9AM2Q 90679729 IC50 = 21877.62 nM T98711 CUDM30 90679730 IC50 = 9772.37 nM T98711 C9PX6B 90679731 IC50 = 1047.13 nM T98711 C1S8AL 91031465 IC50 = 220 nM T98711 CG9JP4 91689645 IC50 = 3600 nM T98711 C7C9RB 91689712 IC50 = 30800 nM T98711 C8NC7S 91689713 IC50 = 32600 nM T98711 CAM0G8 91864546 IC50 = 2.18 nM T98711 CUPK70 91885433 IC50 = 3900 nM T98711 C5RF6O 101077957 IC50 > 30000 nM T98711 C4HLR3 101528287 IC50 > 30000 nM T98711 C20CYQ 101879984 IC50 = 585 nM T98711 C5V2JH 101886788 IC50 = 256 nM T98711 CLO03N 101886789 IC50 = 41.4 nM T98711 CF6EI0 101886790 IC50 = 5.45 nM T98711 C52VTG 101886792 IC50 = 19.1 nM T98711 CV3A0F 101886793 IC50 = 501 nM T98711 CI2U0Y 101886794 IC50 = 197 nM T98711 C56IGC 101886796 IC50 = 258 nM T98711 C6W2JF 101898808 Ki = 16.1 nM T98711 C81WRJ 101910778 IC50 = 4900 nM T98711 CDBZ20 102189779 IC50 = 2844 nM T98711 C1PAK7 102257397 IC50 = 13460 nM T98711 C71RIU 102257398 IC50 = 8930 nM T98711 C4XMG6 102257401 IC50 = 10420 nM T98711 C0NV1I 102286159 IC50 > 10000 nM T98711 C4LJ9O 102369422 IC50 = 267 nM T98711 CY93VO 102369423 IC50 = 328 nM T98711 CYG4M5 102484612 IC50 > 50000 nM T98711 CDRX58 118622604 IC50 > 40000 nM T98711 CP5Z8M 118622610 IC50 = 16200 nM T98711 C7TZ2R 118622611 IC50 = 12700 nM T98711 CRW07P 118622616 IC50 = 8500 nM T98711 CIP1L6 118706200 IC50 = 99 nM T98711 C9M3EL 118709900 IC50 = 765 nM T98711 CMWO04 118709901 IC50 = 228 nM T98711 C39HSZ 118709912 IC50 = 2030 nM T98711 CI38GE 118709913 IC50 = 2380 nM T98711 CH5V0G 118709914 IC50 = 2230 nM T98711 CBP3S5 118709915 IC50 = 12600 nM T98711 CT1J4G 118709916 IC50 = 827 nM T98711 C4IZB0 118709917 IC50 = 1420 nM T98711 C7JDT6 118709918 IC50 = 5620 nM T98711 CEY60K 118709968 IC50 = 286 nM T98711 C8GS0O 118709970 IC50 = 120 nM T98711 CAGS07 118709972 IC50 = 205 nM T98711 C40GLT 118709974 IC50 = 337 nM T98711 C1J0IZ 118711805 Ki = 31.7 nM T98711 C8D5HF 118711806 Ki = 29.8 nM T98711 CLG7K5 118711807 Ki = 34 nM T98711 CQB1O3 118711808 Ki = 32.4 nM T98711 C5C3XE 118711809 Ki = 8.1 nM T98711 C3H2YI 118711810 Ki = 32.5 nM T98711 COUQ50 118711811 Ki = 20.2 nM T98711 COSI80 118711812 Ki = 23.7 nM T98711 CJG10W 118711813 Ki = 23.2 nM T98711 CNH93M 118711814 Ki = 31.2 nM T98711 C2Q8IE 118711815 Ki = 17.5 nM T98711 C3C0QD 118711816 Ki = 20 nM T98711 CG62FL 118711817 Ki = 35 nM T98711 C9U5SV 118712170 Ki = 34.5 nM T98711 C9KUS7 118712171 Ki = 50.9 nM T98711 CJH4K5 118712172 Ki = 37.5 nM T98711 CB74FU 118712173 Ki = 40 nM T98711 C1J5NW 118715681 IC50 = 79900 nM T98711 C2YJB1 118715683 IC50 = 70700 nM T98711 CO98FC 118715684 IC50 = 3020 nM T98711 C0JPI2 118715685 IC50 = 25400 nM T98711 CAI03B 118715686 IC50 = 15900 nM T98711 CVN98D 118715709 IC50 = 32290 nM T98711 CG78ML 118715710 IC50 = 11750 nM T98711 CBO21H 118715711 IC50 = 17420 nM T98711 C5JO1E 118715712 IC50 = 20120 nM T98711 CK8MI7 118715713 IC50 = 10240 nM T98711 C5S7WZ 118715714 IC50 = 26330 nM T98711 CN6QV9 118715715 IC50 = 18470 nM T98711 CF0RX8 118715716 IC50 = 52580 nM T98711 C6MD2K 118715717 IC50 = 10130 nM T98711 C57BFX 118715718 IC50 = 8840 nM T98711 C1EJ5Q 118715719 IC50 = 39650 nM T98711 CQ92DR 118715720 IC50 = 40740 nM T98711 CRD9N0 118715721 IC50 = 279110 nM T98711 C6T0HL 118715722 IC50 = 68250 nM T98711 CQS06R 118715723 IC50 = 41910 nM T98711 C31XUV 118715724 IC50 = 96920 nM T98711 C3ZO6M 118715725 IC50 = 75090 nM T98711 CV98EO 118718831 IC50 = 1800 nM T98711 CLE2S7 118720934 IC50 = 982 nM T98711 C23AHU 118720935 IC50 = 742 nM T98711 CJWC73 118720936 IC50 = 181 nM T98711 CCSQ94 118721626 IC50 = 635 nM T98711 CL7JH8 118721627 IC50 = 14.5 nM T98711 CK2G3V 118721628 IC50 = 1280 nM T98711 CU83LO 118721629 IC50 = 329 nM T98711 CJ3S7L 118721630 IC50 = 970 nM T98711 C4F0TD 118721871 IC50 = 742 nM T98711 C5MR9S 118721872 IC50 = 287 nM T98711 CK85GL 118721873 IC50 = 234 nM T98711 CRTA65 118721874 IC50 = 96.1 nM T98711 C6HM0O 118721875 IC50 = 47.8 nM T98711 C0C6VE 118724841 IC50 = 5080 nM T98711 CHX5E4 118724846 IC50 = 2000 nM T98711 C3MX8I 118724859 IC50 = 930 nM T98711 C5P3GX 118725584 IC50 = 3000 nM T98711 C4N1ZC 118725585 IC50 = 1200 nM T98711 C4SK9H 118725586 IC50 = 7000 nM T98711 CI58BM 118725587 IC50 = 15000 nM T98711 C92JNZ 118725588 IC50 = 61000 nM T98711 CAK26D 118725589 IC50 = 161000 nM T98711 C3OR9J 118725590 IC50 = 210000 nM T98711 C8ZG3S 118727884 IC50 = 550 ug.mL-1 T98711 CXOA52 118730192 IC50 = 5900 nM T98711 C27ZWI 118730193 IC50 = 7100 nM T98711 CEQ56Z 118730194 IC50 = 7300 nM T98711 C3D6VY 118730195 IC50 = 40600 nM T98711 CJ2P9D 118730196 IC50 = 9700 nM T98711 CI2X8N 118730197 IC50 = 31200 nM T98711 C07TJO 118732687 IC50 = 56.3 nM T98711 CFN57B 118732688 IC50 = 5.2 nM T98711 C1UWN7 118732689 IC50 = 10.2 nM T98711 C2LJX1 118732690 IC50 = 20.5 nM T98711 C1GS6P 118732691 IC50 = 19.2 nM T98711 CS73OE 118732692 IC50 = 34.7 nM T98711 C62UPS 118732693 IC50 = 110.1 nM T98711 CNB83Q 118734712 IC50 = 124.32 nM T98711 CX80VO 118734713 IC50 = 112.72 nM T98711 C87YTM 118736706 IC50 > 5000 nM T98711 C4CTX6 118736714 IC50 > 5000 nM T98711 CMB54K 118736716 IC50 > 5000 nM T98711 COS59D 118736718 IC50 > 5000 nM T98711 CIB78Z 118736720 IC50 = 2400 nM T98711 C2PO6M 118736722 IC50 = 3500 nM T98711 C0YHI7 122180159 IC50 > 30000 nM T98711 C5K0RY 122180160 Ki = 4780 nM T98711 C71TKE 122180161 IC50 > 30000 nM T98711 C9QKP3 122180162 IC50 = 420 nM T98711 CQL13W 122180163 IC50 = 1370 nM T98711 CMR72I 122180164 IC50 > 30000 nM T98711 C1X9KB 122180406 IC50 = 950 nM T98711 CMC26Y 122180416 IC50 = 950 nM T98711 CEJ8S0 122180431 IC50 = 890 nM T98711 CKM1E7 122180462 IC50 = 9300 nM T98711 CH36VG 122182060 IC50 = 2140 nM T98711 C4PB1D 122182066 IC50 = 215 nM T98711 CDI8W2 122186374 IC50 = 128740 nM T98711 CK0WP5 122186375 IC50 = 110530 nM T98711 CA7U0N 122186376 IC50 = 187540 nM T98711 CO8V2R 122186377 IC50 = 119210 nM T98711 CE67WU 122186379 IC50 = 118540 nM T98711 C6JYH5 122186381 IC50 = 296530 nM T98711 CLTA13 122186382 IC50 = 105230 nM T98711 C1FKJ5 122186383 IC50 = 106410 nM T98711 C8NRX7 122186486 IC50 = 99740 nM T98711 CMCJ76 122186487 IC50 = 89240 nM T98711 CS5C0T 122186488 IC50 = 151870 nM T98711 C9WA3O 122186489 IC50 = 81410 nM T98711 C8KFR9 122186490 IC50 = 26530 nM T98711 CV4EJ3 122186491 IC50 = 151350 nM T98711 CU08GD 122186492 IC50 = 4520 nM T98711 CI7UZ4 122186493 IC50 = 44830 nM T98711 CKYL61 122186494 IC50 = 5310 nM T98711 CGC6T5 122186495 IC50 = 140930 nM T98711 CDU7H8 122186496 IC50 = 78020 nM T98711 C0JK8P 122186497 IC50 = 491730 nM T98711 C1T7UF 122186498 IC50 = 25910 nM T98711 C21LZX 122186499 IC50 = 187540 nM T98711 CZ38FY 122186500 IC50 = 160950 nM T98711 C8CGX0 122186502 IC50 = 103430 nM T98711 CC28ZL 122186503 IC50 = 167820 nM T98711 CD37LR 122186505 IC50 = 75890 nM T98711 CP4V8H 122191089 IC50 = 1200 nM T98711 C7OGL4 122191091 IC50 = 10000 nM T98711 C73UCL 122191093 IC50 = 20000 nM T98711 C16CXB 122193107 IC50 = 280 nM T98711 C0Q6AY 122193108 IC50 = 340 nM T98711 CM8C5G 122193110 IC50 = 2800 nM T98711 CBQW34 122193112 IC50 = 4100 nM T98711 CAXZ47 122193114 IC50 = 5100 nM T98711 C0ASQ2 122193116 IC50 = 4800 nM T98711 CXN7T8 122193118 IC50 = 5800 nM T98711 CDKJ53 122193120 IC50 = 8900 nM T98711 C6S7CV 122193124 IC50 = 6800 nM T98711 CL8J3Z 122193126 IC50 = 7900 nM T98711 CZ96MQ 122193128 IC50 = 7500 nM T98711 CCZJ35 122193130 IC50 = 80 nM T98711 C7N1BE 122193132 IC50 = 2300 nM T98711 C0FJ1G 122193134 IC50 = 1100 nM T98711 CSU6Q5 122193237 IC50 = 710 nM T98711 CSY2D4 122193239 IC50 = 860 nM T98711 C5VTJ4 122193241 IC50 = 720 nM T98711 C5XAM3 122193243 IC50 = 650 nM T98711 CC7E1R 122194787 IC50 = 1300 nM T98711 CNH49U 122194788 IC50 = 620 nM T98711 CLG31E 122194789 IC50 = 290 nM T98711 CLOD26 122194790 IC50 = 400 nM T98711 CY3EJ9 122194791 IC50 = 690 nM T98711 CI7Q9F 122194792 IC50 = 700 nM T98711 C9C7VG 122194793 IC50 = 1530 nM T98711 C2A4ES 122194881 IC50 = 80 nM T98711 CI2K5Z 122194882 IC50 = 20 nM T98711 C1E3LP 122194883 IC50 = 770 nM T98711 C4A8JM 122194884 IC50 = 90 nM T98711 CR79OE 122194885 IC50 = 130 nM T98711 CZ8L9J 122194886 IC50 = 400 nM T98711 CK7B8R 122194887 IC50 = 700 nM T98711 CSNM01 122194888 IC50 = 54 nM T98711 C5JXL2 122199175 IC50 = 20 nM T98711 CEX9B4 122199179 IC50 = 1400 nM T98711 CPJ2K1 122199184 IC50 = 1900 nM T98711 C3N9DJ 122199186 IC50 = 70 nM T98711 C1T5SW 122199188 IC50 = 1600 nM T98711 CJV5B8 122387041 IC50 = 5000 nM T98711 CI89OZ 122387042 IC50 = 5000 nM T98711 CYWM69 122387043 IC50 = 11000 nM T98711 CFVL05 122387044 IC50 = 38000 nM T98711 CFI4B3 122387045 IC50 = 9600 nM T98711 CNS65E 122387046 IC50 = 11100 nM T98711 C6BG0C 122581932 Ki = 1.71 nM T98711 C50XJY 122581936 IC50 = 4.9 nM T98711 CQ8MG5 122581957 IC50 = 1.03 nM T98711 CO01UP 127025001 IC50 = 2670 nM T98711 CT6H9W 127025002 IC50 = 1680 nM T98711 C2Q8FW 127025129 IC50 = 2800 nM T98711 CAB51G 127025336 IC50 = 15280 nM T98711 CO3NW2 127025337 IC50 = 16250 nM T98711 CHW76D 127025338 IC50 = 12340 nM T98711 C06WQV 127025339 IC50 = 14660 nM T98711 CN4S6W 127025340 IC50 = 13490 nM T98711 C35YFW 127025347 IC50 = 14070 nM T98711 CU5Y2J 127025348 IC50 = 12440 nM T98711 CZNG40 127025349 IC50 = 11870 nM T98711 CQ32HN 127025350 IC50 = 14950 nM T98711 C8HT6M 127025617 IC50 = 2930 nM T98711 CH6A2X 127026192 IC50 = 1980 nM T98711 C2MHZ4 127026193 IC50 = 3450 nM T98711 C71BST 127026245 IC50 = 3800 nM T98711 C5NE2H 127027141 IC50 = 23790 nM T98711 CB25JK 127027142 IC50 = 26600 nM T98711 CT70GX 127027146 IC50 = 6120 nM T98711 CDV42T 127027424 IC50 = 14710 nM T98711 C6M5VF 127027425 IC50 = 15920 nM T98711 CX4YN3 127027643 IC50 = 15.7 nM T98711 C4AE0D 127027644 IC50 = 4.68 nM T98711 CJU4L1 127027645 IC50 = 10.8 nM T98711 CJWO49 127027646 IC50 = 80.6 nM T98711 CD5G9O 127027963 IC50 = 10.2 nM T98711 CBC0Y6 127028241 IC50 = 9000 nM T98711 C6R4EA 127028375 IC50 = 15090 nM T98711 CV5C7L 127028376 IC50 = 26130 nM T98711 C0NC1G 127028377 IC50 = 25420 nM T98711 CTF47Q 127028378 IC50 = 23810 nM T98711 CCO6D4 127028379 IC50 = 26040 nM T98711 C3DGN9 127029030 IC50 = 4900 nM T98711 C3FHL4 127029354 IC50 = 9100 nM T98711 CWJ80N 127029355 IC50 = 40000 nM T98711 C9RD5O 127029356 IC50 = 19300 nM T98711 C3BOU8 127029357 IC50 = 5700 nM T98711 C1QL4R 127033914 IC50 = 13 nM T98711 CF3HK1 127034304 IC50 > 200000 nM T98711 CY1I9K 127034570 IC50 = 163800 nM T98711 CZ3EV8 127035309 IC50 = 1.23 nM T98711 C7TQI5 127035310 IC50 = 8.89 nM T98711 C4HJR5 127036051 IC50 = 30 nM T98711 CKUR62 127036052 IC50 = 6.9 nM T98711 C1XE2Y 127036053 IC50 = 11.6 nM T98711 CF19QE 127036054 IC50 = 26.1 nM T98711 C07GWU 127036055 IC50 = 7.35 nM T98711 CA3MW8 127036212 IC50 = 31.9 nM T98711 COZ7S8 127036213 IC50 = 2.48 nM T98711 CW5MQ7 127036214 IC50 = 1.3 nM T98711 CPY5X2 127036215 IC50 = 0.49 nM T98711 C4JFN8 127036216 IC50 = 2.54 nM T98711 CX85YQ 127036232 IC50 = 2.3 nM T98711 CS6ND0 127036233 IC50 = 0.48 nM T98711 CVO6Y9 127036234 IC50 = 2.35 nM T98711 C1WLH2 127036472 IC50 = 30.9 nM T98711 C59WQJ 127036580 IC50 = 33.33 ug.mL-1 T98711 CM73TG 127036581 IC50 > 80 ug.mL-1 T98711 C65EVQ 127036864 IC50 = 8100 nM T98711 C0RXJ6 127036990 IC50 = 7900 nM T98711 C2LH5V 127037240 IC50 = 12.8 nM T98711 CH63BP 127037241 IC50 = 6.86 nM T98711 CIHE05 127037242 IC50 = 17.9 nM T98711 CG02IX 127037256 IC50 > 80 ug.mL-1 T98711 CMI6G3 127037257 IC50 = 66.67 ug.mL-1 T98711 C8S5LU 127037259 IC50 > 80 ug.mL-1 T98711 C8AYT1 127037384 IC50 = 4.87 nM T98711 C49PET 127037401 IC50 = 77 ug.mL-1 T98711 CUYD86 127037417 IC50 = 39.6 ug.mL-1 T98711 C3SN7K 127037516 IC50 > 80 ug.mL-1 T98711 CD16UI 127037518 IC50 > 80 ug.mL-1 T98711 CHR89X 127037869 IC50 = 16840 nM T98711 C0RTX1 127038878 IC50 = 24670 nM T98711 CO81HM 127038907 IC50 = 23770 nM T98711 C4QWS0 127043654 IC50 = 1030000 nM T98711 CQZW98 127043697 IC50 = 0.28 nM T98711 CCGN43 127043698 IC50 = 0.53 nM T98711 C7XP8D 127043699 IC50 = 1.17 nM T98711 CCRX05 127043700 IC50 = 42.7 nM T98711 C5IQU4 127043705 IC50 = 78.2 nM T98711 C09KSX 127043865 IC50 = 32.1 nM T98711 CG3DR4 127043866 IC50 = 2.85 nM T98711 CCWJ60 127043867 IC50 = 1.23 nM T98711 CG20QN 127043868 IC50 = 0.79 nM T98711 C3W8MB 127043871 IC50 = 15.9 nM T98711 C9M0KG 127043877 IC50 = 1230 nM T98711 CZA3R7 127043878 IC50 = 15.2 nM T98711 CX1G8L 127043879 IC50 = 122000 nM T98711 C54WIK 127043880 IC50 = 71.2 nM T98711 CP72LZ 127044176 IC50 = 0.27 nM T98711 C2VJ7H 127044293 IC50 = 400000 nM T98711 CF9BD1 127044471 IC50 = 1190000 nM T98711 C5GVQ3 127044472 IC50 = 800000 nM T98711 CT6YL4 127044473 IC50 = 400000 nM T98711 C7S5KZ 127044474 IC50 = 310000 nM T98711 CXS8Z2 127044620 IC50 = 900000 nM T98711 CS0CG7 127044621 IC50 = 8100 nM T98711 CI21OB 127044622 IC50 = 2000 nM T98711 C3PB5G 127044623 IC50 = 590 nM T98711 CXN83I 127044654 IC50 = 2.06 nM T98711 C97PFW 127044655 IC50 = 1.3 nM T98711 CC7W8O 127044656 IC50 = 1.15 nM T98711 C19MEI 127044657 IC50 = 3.51 nM T98711 CMU0Q3 127045144 IC50 = 1.44 nM T98711 CZOJ81 127045292 IC50 = 2.75 nM T98711 C37IKG 127045293 IC50 = 1.19 nM T98711 C8V2DN 127048404 IC50 = 1440 nM T98711 CQ16RS 127048405 IC50 = 669 nM T98711 CY71LG 127048406 IC50 = 7510 nM T98711 CW2B3M 127048716 IC50 = 784 nM T98711 CKEN30 127048749 IC50 = 1220 nM T98711 C23EOB 127049071 IC50 = 690 nM T98711 CU8I7J 127049072 IC50 = 988 nM T98711 C23YAL 127049073 IC50 = 245 nM T98711 C2BVI5 127049123 IC50 = 850 nM T98711 CG65ES 127049124 IC50 = 1400 nM T98711 CR39WO 127049125 IC50 = 290 nM T98711 C7X0IE 127049126 IC50 = 1060 nM T98711 CU85GC 127049730 IC50 = 76 nM T98711 CRW64G 127049731 IC50 = 3240 nM T98711 CXB9K4 127050511 IC50 = 950 nM T98711 CCI4E1 127050512 IC50 = 1420 nM T98711 CZGX21 127050513 IC50 = 1030 nM T98711 CS8X7B 127050845 IC50 = 2210 nM T98711 CRE9O5 127051536 IC50 = 286 nM T98711 C39VRD 127051623 IC50 = 400 nM T98711 C5CYS7 127051624 IC50 = 3010 nM T98711 CN63WP 129766223 IC50 = 520 nM T98711 CYQT64 129904916 IC50 > 100000 nM T98711 C3OH2U 132281442 IC50 = 68.2 nM T98711 CZ2JQ4 132427688 IC50 = 260 nM T98711 C61DGH 132495293 IC50 = 1020 nM T98711 C5AU1H 132495295 IC50 = 5270 nM T98711 CZ3OD0 132495360 IC50 = 2600 nM T98711 CBN5C0 132495361 IC50 = 127 nM T98711 CM7PY1 132547201 Ki = 160 nM T98711 C3F4ME 132569621 IC50 = 7300 nM T98711 CX59ME 133561407 IC50 > 10000 nM T98711 C4YH6G 134129916 IC50 = 25400 nM T98711 C0EU7L 134130629 IC50 = 6350 nM T98711 C5Z9WG 134131252 IC50 = 29.7 nM T98711 C8R7KL 134131932 IC50 = 52.44 nM T98711 CCJF74 134132255 IC50 = 39 nM T98711 C3VO0S 134132482 IC50 = 8 nM T98711 C9UGN0 134132984 IC50 = 37 nM T98711 CA5BJ4 134133150 IC50 = 6.4 nM T98711 C6VS5U 134133379 IC50 = 137 nM T98711 CVF3T5 134133384 IC50 = 30 nM T98711 CZTV48 134134429 IC50 = 4370 nM T98711 CYB1T5 134134557 IC50 = 30.41 nM T98711 CB31IT 134134606 IC50 = 8550 nM T98711 CYWV57 134134625 IC50 > 10000 nM T98711 C71IYO 134135593 IC50 = 15 nM T98711 CP1E5Y 134135669 IC50 = 3.79 nM T98711 CB19DO 134135810 IC50 = 65 nM T98711 CZ9YA3 134135893 IC50 = 7360 nM T98711 C9OE5Y 134135942 IC50 = 760 nM T98711 C8X1DP 134136230 IC50 = 5 nM T98711 CHB06R 134136355 IC50 = 41400 nM T98711 CP3RN6 134136543 IC50 = 1020 nM T98711 CK06MI 134136825 IC50 = 49200 nM T98711 CM83OH 134137000 IC50 = 1910 nM T98711 C7XE0G 134137541 IC50 = 5120 nM T98711 CSA09I 134137557 IC50 = 79 nM T98711 C97CUD 134137716 IC50 = 64 nM T98711 CYG95X 134137746 IC50 = 18800 nM T98711 C9JW0A 134137761 IC50 = 6080 nM T98711 CZB2H1 134137882 IC50 = 73 nM T98711 C3MFB4 134138158 IC50 = 3.59 nM T98711 C3WL0X 134138347 IC50 = 5600 nM T98711 CTQY30 134138725 IC50 = 37400 nM T98711 C5B6YK 134138931 IC50 = 43 nM T98711 CYR2D1 134138980 IC50 = 48.13 nM T98711 CQU8T5 134139124 IC50 = 281 nM T98711 C32PAF 134139263 IC50 > 200000 nM T98711 C6BH1E 134139570 IC50 = 12 nM T98711 CM5D2F 134139579 IC50 = 65700 nM T98711 C5E6PV 134139682 IC50 = 42 nM T98711 C0VGT1 134140048 IC50 = 5000 nM T98711 COB3U4 134140335 IC50 = 4370 nM T98711 C1A7EP 134140534 IC50 = 570 nM T98711 CBS53R 134140571 IC50 = 4.12 nM T98711 CH2W1P 134140732 IC50 = 6 nM T98711 C73LGF 134140781 IC50 = 8641 nM T98711 CU2H9S 134140801 IC50 = 6.97 nM T98711 CYW3P5 134141480 IC50 = 53.76 nM T98711 C6NCM8 134141704 IC50 = 10 nM T98711 CC6P0J 134141898 IC50 = 38900 nM T98711 CHDC50 134142324 IC50 = 15 nM T98711 CSYM31 134142478 IC50 = 23444 nM T98711 CUP09Q 134142596 IC50 = 4390 nM T98711 C9L1VS 134142725 IC50 = 1560 nM T98711 CI38NM 134143999 IC50 = 2870 nM T98711 C47KWL 134144584 IC50 = 4040 nM T98711 CIE6T7 134144753 IC50 = 21 nM T98711 CZ4WL3 134144932 IC50 = 365 nM T98711 CKAF58 134145123 IC50 = 15 nM T98711 C4Z9HA 134145445 IC50 = 30 nM T98711 CP0D4F 134146126 IC50 = 1223 nM T98711 CZVL70 134146128 IC50 = 12800 nM T98711 C89RCM 134146339 IC50 = 78700 nM T98711 C1K2XO 134146719 IC50 = 2520 nM T98711 CZM9O4 134146757 IC50 = 5890 nM T98711 CBOY65 134146798 IC50 = 24 nM T98711 CW1U8M 134147085 IC50 = 3370 nM T98711 CID47M 134147264 IC50 = 7 nM T98711 C3G2FL 134147416 IC50 = 47.33 nM T98711 CNVG70 134147548 IC50 > 10000 nM T98711 C5A1SG 134147628 IC50 = 1420 nM T98711 C5E6RH 134147648 IC50 > 10000 nM T98711 CE7X9I 134148653 IC50 = 7 nM T98711 CXOD70 134148863 IC50 = 32.07 nM T98711 C7E3YA 134149382 IC50 > 10000 nM T98711 C03PFN 134149524 IC50 = 3930 nM T98711 CSMP25 134149784 IC50 = 3060 nM T98711 C4Y5ZX 134150471 IC50 = 260 nM T98711 CRZ2W4 134150858 IC50 = 3306 nM T98711 C5BMP0 134151164 IC50 = 456.21 nM T98711 C4RD1Z 134151725 IC50 = 22.56 nM T98711 CJ98WY 134152913 IC50 = 6400 nM T98711 CIV53R 134153098 IC50 = 11.58 nM T98711 CE0DW1 134153138 IC50 = 4480 nM T98711 CA2KR0 134153338 IC50 = 2 nM T98711 CT51CQ 134153533 IC50 = 13 nM T98711 CPBG73 134153558 IC50 = 4590 nM T98711 CNC58Z 134154903 IC50 = 9 nM T98711 CO8IQ0 134155051 IC50 = 1.8 nM T98711 C9QXG2 134155279 IC50 = 23 nM T98711 CA59GH 134155309 IC50 = 75 nM T98711 CJ7Y1Q 134155675 IC50 = 50200 nM T98711 CQA14Y 134155772 IC50 = 384 nM T98711 CL80HA 134155833 IC50 = 13 nM T98711 CPBJ79 134155988 IC50 = 76900 nM T98711 CS3X9K 134156217 IC50 = 29 nM T98711 CC84RT 134157228 IC50 = 2190 nM T98711 CC0IG7 134157232 IC50 = 54396 nM T98711 CW4H7K 134157259 IC50 = 8 nM T98711 CT0IZ2 134157388 IC50 = 77 nM T98711 CY65KP 134157669 IC50 = 11 nM T98711 CJS28R 134157781 IC50 = 18 nM T98711 CUD08L 134817200 IC50 = 1690 nM T98711 CEW6B4 135401162 IC50 = 4000 nM T98711 CQ0WB8 135409581 IC50 > 50000 nM T98711 CXS6M1 135410029 Ki = 390000 nM T98711 C6SMT5 135517369 IC50 = 2200 nM T98711 C5ZCK6 135531254 IC50 > 50000 nM T98711 C8TQ1R 135595416 IC50 = 16000 nM T98711 C73ZKR 135599085 IC50 = 2500 nM T98711 C5YH3F 135621406 IC50 = 194 nM T98711 CFNX32 135777608 Ki = 212400 nM T98711 C98KNJ 135846078 IC50 > 10000 nM T98711 C81ITK 135846093 IC50 > 10000 nM T98711 C8I1WV 135905682 IC50 = 14000 nM T98711 CC2L8T 136044207 IC50 = 13700 nM T98711 CQSW91 136110931 IC50 = 140220 nM T98711 CB1ZV3 136110932 IC50 = 101520 nM T98711 CZ8UM3 136239360 IC50 = 3310 nM T98711 C4TR7Z 136239361 IC50 = 57810 nM T98711 CW2NC0 136239465 Ki = 446480 nM T98711 C92YAW 136239487 IC50 = 231610 nM T98711 CO1TR8 136242439 IC50 = 23000 nM T98711 CL0W4D 136244480 IC50 = 58250 nM T98711 CW4LE8 136244481 IC50 = 358 nM T98711 CKCE30 136244497 IC50 = 8810 nM T98711 CU5VF2 136244586 IC50 = 56810 nM T98711 CV3ST2 136254438 IC50 = 38510 nM T98711 CNG5M3 136254439 IC50 = 75410 nM T98711 CH29ZJ 136254440 IC50 = 8110 nM T98711 CYD96O 136254441 IC50 = 116610 nM T98711 C86MBG 136260466 IC50 = 136910 nM T98711 CKC84W 136260526 IC50 = 57110 nM T98711 CVE2S8 136260527 IC50 = 68410 nM T98711 C1X8GA 136260528 IC50 = 56510 nM T98711 CJZ38F 136264303 IC50 = 64320 nM T98711 C7CGQ4 136264469 IC50 = 52140 nM T98711 COQ2J8 136264470 IC50 = 19370 nM T98711 C5CB7E 136268789 IC50 > 50000 nM T98711 CEBX51 136498868 IC50 = 3970 nM T98711 CYM59N 136498869 IC50 = 4700 nM T98711 C8BAP5 137125243 IC50 = 24100 nM T98711 C8T1NA 137169079 IC50 > 50000 nM T98711 CEL8Q2 137631614 IC50 = 4780 nM T98711 CRH92A 137632694 IC50 = 18 nM T98711 CX6YO4 137632785 IC50 > 5000 nM T98711 CG21YK 137632803 IC50 = 20020 nM T98711 CIY0P1 137632867 IC50 = 400 nM T98711 CQE2C5 137633051 IC50 = 300 nM T98711 C8FSZ4 137633176 IC50 > 5000 nM T98711 CC3Z7H 137633188 IC50 = 40950 nM T98711 C0Y2FZ 137633400 IC50 = 9910 nM T98711 CVK1Z4 137633425 IC50 = 22150 nM T98711 C02GNF 137633542 IC50 = 410 nM T98711 CEI0T6 137633782 IC50 = 14600 nM T98711 C9QLT1 137633879 IC50 = 5690 nM T98711 CCF19I 137634197 IC50 = 50 nM T98711 CVK63S 137634258 IC50 = 3500 nM T98711 C0T9ZD 137634437 IC50 = 3830 nM T98711 CXDY28 137634711 IC50 > 50000 nM T98711 CUSI50 137634757 IC50 > 5000 nM T98711 CH2IJ8 137634974 IC50 = 9100 nM T98711 CU0DK7 137635136 IC50 = 9800 nM T98711 CJ21RK 137635381 IC50 = 390 nM T98711 C7S9TN 137635450 IC50 = 1100 nM T98711 CF08CP 137635497 IC50 = 376710 nM T98711 CK12JV 137635625 IC50 = 230 nM T98711 C82ELC 137635812 IC50 = 82000 nM T98711 C1GT8Y 137635839 IC50 = 302450 nM T98711 C9GA2C 137635913 IC50 = 1584.89 nM T98711 CWSF64 137636375 IC50 = 54100 nM T98711 CV8W7S 137637059 IC50 > 50000 nM T98711 C2WBP4 137637064 IC50 = 3200 nM T98711 C2Z5KH 137637592 IC50 = 6720 nM T98711 CZ5WE1 137637732 IC50 > 50000 nM T98711 CWB7O3 137637856 IC50 = 55 nM T98711 CFP1G9 137637896 IC50 = 11460 nM T98711 CFI74R 137637910 IC50 = 3600 nM T98711 C07FMS 137638163 IC50 > 5000 nM T98711 CC7E4I 137638765 IC50 > 50000 nM T98711 CR5G9J 137638769 IC50 = 1600 nM T98711 CJP8W9 137638885 IC50 = 74250 nM T98711 C4AX5H 137639047 IC50 = 12900 nM T98711 C6DJ8C 137639617 IC50 = 2230 nM T98711 C89ELW 137639718 IC50 = 10200 nM T98711 CRG16O 137639776 IC50 = 11380 nM T98711 CJ1L2M 137639795 IC50 = 150 nM T98711 CPK5O7 137639919 IC50 > 5000 nM T98711 C7EN5K 137640663 IC50 = 10100 nM T98711 CLS48N 137641195 IC50 = 97000 nM T98711 CJ1V3P 137641233 IC50 = 4840 nM T98711 CY5NR3 137641257 IC50 > 50000 nM T98711 CTR8E0 137641522 IC50 = 5011.87 nM T98711 CXL6G5 137641793 IC50 = 8470 nM T98711 CED9V8 137641985 IC50 = 1700 nM T98711 CDY1X7 137641989 IC50 = 20580 nM T98711 CH8B5Q 137642077 IC50 = 7140 nM T98711 C3EL4I 137642431 IC50 = 5600 nM T98711 C6BZ2P 137642547 IC50 = 5490 nM T98711 CH2A8I 137642953 IC50 = 11670 nM T98711 CT72VS 137643173 IC50 > 5000 nM T98711 C15JOE 137643788 IC50 = 5900 nM T98711 C49CZB 137643848 IC50 > 5000 nM T98711 C9B2ZE 137644072 IC50 = 71000 nM T98711 CM2CG5 137644485 IC50 = 286720 nM T98711 C5OEB2 137644607 IC50 > 5000 nM T98711 C4YGM1 137644680 IC50 > 5000 nM T98711 CM91SH 137644867 IC50 = 13050 nM T98711 C7TWP1 137644997 IC50 = 8900 nM T98711 CSCI58 137645198 IC50 = 10410 nM T98711 C1DHM4 137645326 IC50 = 8200 nM T98711 CG96IN 137645336 IC50 = 5710 nM T98711 CAOM59 137645444 IC50 = 12970 nM T98711 C4OQ9U 137645703 IC50 = 6100 nM T98711 CC2SY8 137646193 IC50 > 50000 nM T98711 CPV4Z7 137646357 IC50 = 25900 nM T98711 C5CPS2 137646394 Ki = 0.0111 nM T98711 CAGB15 137646401 IC50 = 3800 nM T98711 CV0I6J 137647059 IC50 = 14190 nM T98711 CL45YE 137647453 IC50 = 2990 nM T98711 C9J3XC 137647729 IC50 = 5000 nM T98711 CO3P1M 137647800 IC50 = 22680 nM T98711 CNUC94 137647812 IC50 = 110000 nM T98711 C5MJG7 137647822 IC50 = 1000 nM T98711 C0ZXC8 137647877 IC50 = 300 nM T98711 C41KDG 137648030 IC50 > 50000 nM T98711 CEC78J 137648049 IC50 = 70 nM T98711 CJP1G6 137648183 IC50 = 30400 nM T98711 CC5R7U 137648202 IC50 = 9600 nM T98711 CBPK31 137648694 IC50 = 2511.89 nM T98711 C07ZJU 137648924 IC50 = 16880 nM T98711 CMRI71 137649149 IC50 = 2300 nM T98711 CW2UK0 137649211 IC50 = 8600 nM T98711 C30VHY 137649676 IC50 = 145690 nM T98711 C6JEQ0 137649792 IC50 = 1350 nM T98711 C7Z4MI 137649813 IC50 = 14000 nM T98711 C12HUM 137650006 IC50 = 25000 nM T98711 CBFM14 137650067 IC50 > 10000 nM T98711 C0ZM5Q 137650571 IC50 = 632 nM T98711 CH50RP 137650702 IC50 = 1200 nM T98711 CHW83L 137650736 IC50 = 67 nM T98711 CJW29P 137650881 IC50 = 3800 nM T98711 C54VBE 137651033 IC50 = 2760 nM T98711 CTOX45 137651149 IC50 = 1437 nM T98711 CXM65D 137651291 IC50 = 110000 nM T98711 CWQ87J 137651676 IC50 = 702 nM T98711 C3WL9S 137652298 IC50 = 1850 nM T98711 CW9HL2 137652394 IC50 = 360 nM T98711 C1KSJ8 137652783 IC50 = 4780 nM T98711 CHWO15 137652896 IC50 = 7800 nM T98711 CMP3S2 137652915 IC50 = 1560 nM T98711 CQJ78X 137653099 IC50 = 4860 nM T98711 CFPV35 137653376 IC50 = 2340 nM T98711 CSO97E 137653574 IC50 = 4500 nM T98711 CG3V4T 137653648 IC50 = 1200 nM T98711 C6O0AJ 137653712 IC50 = 9700 nM T98711 CX4AM2 137653862 IC50 = 5760 nM T98711 CB1I0V 137654237 IC50 = 23280 nM T98711 C0UNA5 137654399 IC50 = 9500 nM T98711 C0C5OB 137654571 IC50 = 50118.72 nM T98711 C0LR3F 137654627 IC50 > 50000 nM T98711 CO25BH 137654740 IC50 > 5000 nM T98711 CT1PA9 137654741 IC50 = 1300 nM T98711 C58UJM 137654765 IC50 = 41760 nM T98711 C4UZ6L 137654824 IC50 = 7.28 nM T98711 CAQ92O 137654935 IC50 > 5000 nM T98711 CP3R6K 137655004 IC50 = 8900 nM T98711 CS7G0V 137655713 IC50 = 3100 nM T98711 CCA96J 137655921 IC50 = 2200 nM T98711 CMA9P4 137655981 IC50 > 50000 nM T98711 C4XM2Y 137657255 IC50 > 5000 nM T98711 CA26MD 137657287 IC50 = 2500 nM T98711 C61BAH 137657694 IC50 = 25070 nM T98711 CJNL70 137657810 IC50 = 3980 nM T98711 C9XPC4 137657910 IC50 = 17600 nM T98711 CU4B0Q 137658210 IC50 = 170 nM T98711 CT51VW 137658213 IC50 = 24900 nM T98711 CN0SF1 137658402 IC50 = 2140 nM T98711 CW2I9D 137658492 IC50 = 3630 nM T98711 C15GDM 137658514 IC50 = 12080 nM T98711 CQC6G7 137658542 IC50 = 5700 nM T98711 CJU20M 137658706 IC50 = 1300 nM T98711 CC7V1S 137658749 IC50 = 5450 nM T98711 CEV12H 137659101 IC50 = 8800 nM T98711 COL58K 137659202 IC50 = 29800 nM T98711 CSP06U 137659306 IC50 = 29800 nM T98711 CC65MS 137659483 IC50 = 30500 nM T98711 CBD24K 137660365 IC50 = 15800 nM T98711 C8IW5O 137660695 IC50 > 5000 nM T98711 CH34LO 137660979 IC50 = 4030 nM T98711 CKMC76 137661029 IC50 = 12680 nM T98711 C6F7QS 137661135 IC50 = 7.12 nM T98711 C31MDX 137661164 IC50 > 50000 nM T98711 C7E2OH 137661175 IC50 > 5000 nM T98711 CD8W3T 137661581 IC50 = 38.24 nM T98711 C7FL2W 137661647 IC50 = 8400 nM T98711 CQV79Z 137661668 IC50 > 50000 nM T98711 CIJ43L 137662097 IC50 = 263110 nM T98711 C9J4DH 138320049 IC50 = 254 nM T98711 CU3VY8 141700626 IC50 = 2100 nM T98711 CY20TH 141700627 IC50 = 0.26 nM T98711 CC50YG 141700631 IC50 = 230 nM T98711 CU7SJ0 145722355 IC50 = 2.5 nM T98711 C80HQW 145949396 IC50 = 5680 nM T98711 CZ0IR5 145949784 IC50 = 1560 nM T98711 CU15AO 145950308 IC50 = 8410 nM T98711 C3GNZ9 145950384 IC50 = 511 nM T98711 CFU46Z 145950418 IC50 = 310 nM T98711 CN1MF4 145950493 IC50 = 3190 nM T98711 C35CUT 145950652 IC50 = 1270 nM T98711 CQWI16 145950841 IC50 = 356 nM T98711 CN4C6I 145951178 IC50 > 10000 nM T98711 C81CRX 145951391 IC50 = 5270 nM T98711 CSU4Y2 145951896 IC50 = 6540 nM T98711 CL1TK4 145952378 IC50 = 47210 nM T98711 CR26YA 145952393 IC50 = 630 nM T98711 C6VLZ8 145952662 IC50 = 3690 nM T98711 CY7RD4 145953155 IC50 = 378 nM T98711 C2SFL4 145953212 IC50 = 37500 nM T98711 C5U8LK 145953230 IC50 = 4020 nM T98711 C9ZPF5 145954333 IC50 = 372 nM T98711 CP8L3U 145954454 IC50 = 452 nM T98711 CB2PU4 145954736 IC50 = 340 nM T98711 C8LJV7 145954769 IC50 = 1110 nM T98711 CF09RS 145954786 IC50 = 510 nM T98711 CRP68J 145955177 IC50 = 2650 nM T98711 CMYF60 145956446 IC50 = 11700 nM T98711 CRTG06 145956559 IC50 = 3470 nM T98711 CNIR29 145956699 IC50 = 4010 nM T98711 C0Q3MP 145957027 IC50 = 650 nM T98711 C7BY3Q 145957085 IC50 = 2680 nM T98711 COR92I 145957306 IC50 = 9960 nM T98711 CW1M4Y 145958077 IC50 = 4590 nM T98711 C7UK4Q 145958135 IC50 = 990 nM T98711 CG6D8I 145958306 IC50 > 10000 nM T98711 CCBO90 145958532 IC50 > 10000 nM T98711 CTCE08 145958953 IC50 = 25800 nM T98711 C7E0WG 145959287 IC50 = 828 nM T98711 CNS69M 145959783 IC50 > 10000 nM T98711 CLP6E5 145959857 IC50 = 14930 nM T98711 CFUJ38 145959883 IC50 = 10000 nM T98711 CRD76Q 145963428 IC50 = 32530 nM T98711 CD6K7P 145963526 IC50 = 4700 nM T98711 C37BNF 145963787 IC50 = 37.2 nM T98711 CTH70Y 145963788 IC50 = 8320 nM T98711 C85ZOK 145963821 IC50 = 1320 nM T98711 C8VFP2 145963831 IC50 = 20.7 nM T98711 CIZ2D6 145964146 IC50 = 408 nM T98711 CUY37P 145964192 IC50 = 1186 nM T98711 CL8IM7 145964214 IC50 = 3340 nM T98711 CCX4G7 145964403 IC50 = 16.6 nM T98711 C7O1VM 145964717 IC50 = 1001 nM T98711 CC65HS 145965070 IC50 = 12.4 nM T98711 C52IFK 145965199 IC50 = 577 nM T98711 CO09TS 145966146 IC50 = 107 nM T98711 CZ20XJ 145967112 IC50 = 12400 nM T98711 CCVM34 145967131 IC50 = 3720 nM T98711 C4RFE9 145967436 IC50 = 2400 nM T98711 C4CGL8 145968916 IC50 = 4.35 nM T98711 C7NB8L 145970781 IC50 = 103 nM T98711 C8IRS3 145970790 IC50 = 4950 nM T98711 CNS36B 145971232 IC50 = 1750 nM T98711 CS52IM 145971379 IC50 = 48.8 nM T98711 CS2NH6 145971450 IC50 = 154000 nM T98711 CKP39X 145971650 IC50 = 1080 nM T98711 C0RV3Z 145972056 IC50 = 1190 nM T98711 C10KGM 145972388 IC50 = 1030 nM T98711 CADI36 145972622 IC50 = 1290 nM T98711 CVG37T 145972858 IC50 = 26.8 nM T98711 CC3K4N 145972893 IC50 = 8860 nM T98711 CMB59C 145972994 IC50 = 1460 nM T98711 CHA90Q 145973001 IC50 = 145 nM T98711 CE9U6I 145973015 IC50 = 83.3 nM T98711 C8X5YT 145973525 IC50 = 8010 nM T98711 CR01XP 145973666 IC50 = 674 nM T98711 CV2I6R 145973676 IC50 = 950 nM T98711 CP3W4L 145974148 IC50 = 3120 nM T98711 C7WRK1 145974265 IC50 = 7740 nM T98711 CUD2Z0 145974298 IC50 = 45500 nM T98711 C9KNC3 145974491 IC50 = 13400 nM T98711 C2CSU4 145974513 IC50 = 10.5 nM T98711 C8VZ5F 145974561 IC50 > 10000 nM T98711 CJ51HA 145974740 IC50 = 81.5 nM T98711 C5UZ8W 145974825 IC50 = 507 nM T98711 CXS48G 145974962 IC50 = 49300 nM T98711 C80VLM 145975022 IC50 = 107 nM T98711 C26ZBO 145975126 IC50 = 6160 nM T98711 CU2ES3 145975561 IC50 = 45.7 nM T98711 CU1NO6 145976650 IC50 = 280 nM T98711 CEXP52 145976876 IC50 = 16600 nM T98711 CRAM60 145977029 IC50 = 1050 nM T98711 CF4A0B 145977178 IC50 = 2.35 nM T98711 CBFC12 145977206 IC50 = 2030 nM T98711 CEO72I 145977249 IC50 = 29.9 nM T98711 COSM78 145977433 IC50 = 16.3 nM T98711 CL9HU4 145977623 IC50 = 108 nM T98711 CKO6P0 145977734 IC50 = 4320 nM T98711 C2UVJ5 145977785 IC50 = 1210 nM T98711 CYW3U1 145978073 IC50 = 58.9 nM T98711 CUD60Z 145978446 IC50 = 823 nM T98711 CQ6TB5 145978697 IC50 = 37200 nM T98711 CE07DW 145978744 IC50 = 1280 nM T98711 CHX28E 145978908 IC50 = 10300 nM T98711 CZG8R6 145979011 IC50 = 210 nM T98711 C9RQ7P 145979084 IC50 = 670 nM T98711 CXD4H1 145979225 IC50 = 6916.4 nM T98711 CJYX43 145979238 IC50 = 9.5 nM T98711 CGWB38 145979348 Ki = 187000 nM T98711 C7XLF0 145979801 IC50 = 4.571 nM T98711 CX2RW9 145979866 IC50 = 19560 nM T98711 C1D9ZU 145979972 IC50 > 10000 nM T98711 CE0DG7 145980262 IC50 = 265.8 nM T98711 C6PL4V 145980390 IC50 = 1949.84 nM T98711 CW93VH 145980588 IC50 > 10000 nM T98711 CK59PS 145980980 IC50 = 237 nM T98711 CSNL80 145981760 IC50 = 21.8 nM T98711 C8TP1V 145981823 IC50 > 10000 nM T98711 CE84KA 145981976 Ki = 195000 nM T98711 CX3M9J 145981988 IC50 = 4440 nM T98711 CLD9H6 145982286 IC50 = 28 nM T98711 CWNB08 145982383 IC50 = 4250 nM T98711 CFNJ87 145982457 IC50 = 9300 nM T98711 C7VJ1L 145983695 IC50 = 23600 nM T98711 C53SFP 145984170 IC50 = 634.5 nM T98711 CW4X2T 145984359 IC50 > 10000 nM T98711 CSYF87 145984930 IC50 = 103.1 nM T98711 C19IWK 145986527 IC50 = 450 nM T98711 CD73AY 145986601 IC50 = 8790 nM T98711 CCWA30 145986676 IC50 = 20000 nM T98711 CS1CL3 145986706 IC50 = 200 nM T98711 CGLW18 145987198 Ki = 273000 nM T98711 CBG81P 145987259 Ki = 294000 nM T98711 C21BYI 145987407 IC50 = 4300 nM T98711 CAXH94 145987711 IC50 = 28 nM T98711 CJP7H5 145987783 IC50 = 100 nM T98711 C98DHT 145987800 IC50 > 10000 nM T98711 CA82TF 145987838 IC50 = 5800 nM T98711 CLGS98 145988032 IC50 > 10000 nM T98711 C3M1ZO 145988042 IC50 > 10000 nM T98711 CA45JZ 145988111 IC50 = 263.03 nM T98711 C1XU7P 145988798 IC50 > 10000 nM T98711 C2A8MY 145989254 IC50 = 39300 nM T98711 CLG23Y 145989395 IC50 = 20951.3 nM T98711 C6RB3V 145989629 IC50 > 10000 nM T98711 C5BFR8 145989798 IC50 = 19 nM T98711 C6QRA9 145989946 IC50 = 7420 nM T98711 C4OAU8 145989956 IC50 > 10000 nM T98711 CVBP12 145989988 IC50 > 10000 nM T98711 C9NTF8 145990243 IC50 > 10000 nM T98711 C63USF 145990366 Ki = 265000 nM T98711 CDBW68 145990442 IC50 = 9610 nM T98711 C4N1WB 145990478 IC50 = 1.82 nM T98711 CGP60E 145990565 IC50 = 6300 nM T98711 CR59TZ 145990611 IC50 = 9900 nM T98711 CQ4R9F 145990749 IC50 = 84810 nM T98711 CCAM14 145990761 IC50 = 74240 nM T98711 C5QZJ4 145990784 IC50 > 10000 nM T98711 C6AZ2B 145990932 IC50 = 228.6 nM T98711 CK9Z4O 145991455 IC50 = 135 nM T98711 CKQ9N2 145991501 IC50 = 11300 nM T98711 C1ZQ0W 145991508 IC50 = 1570 nM T98711 CQD5J2 145991584 IC50 = 460.4 nM T98711 C1P4MD 145991603 IC50 = 48.1 nM T98711 C8KUE6 145991747 IC50 = 610 nM T98711 CR69KG 145992024 IC50 = 51 nM T98711 C1O3VK 145992136 IC50 = 9310 nM T98711 C84LNF 145992210 Ki = 140000 nM T98711 CB9P8D 145992212 IC50 > 10000 nM T98711 C1WI3A 145992723 IC50 > 10000 nM T98711 C7WA5I 145992788 IC50 = 9 nM T98711 CPBJ68 145992936 IC50 > 10000 nM T98711 CF36AC 145993120 IC50 = 5090 nM T98711 CBK49L 145993204 IC50 = 71 nM T98711 C1FBD7 145993205 IC50 = 150 nM T98711 C5YMR4 145993208 IC50 = 6500 nM T98711 CI9T7A 145993228 IC50 = 1611.8 nM T98711 CNDI85 145993235 IC50 = 2485.1 nM T98711 CQ61NL 145993296 IC50 = 7823 nM T98711 CY2N1D 145993326 IC50 = 4320 nM T98711 CUVC73 145993378 IC50 > 10000 nM T98711 CK54FE 145993438 IC50 > 10000 nM T98711 C30CMY 145993498 IC50 > 10000 nM T98711 C27FDC 145993580 IC50 > 10000 nM T98711 CQ9HB3 145993722 IC50 = 2.29 nM T98711 CY62QA 145993943 Ki = 1.09 nM T98711 CQEN91 145993998 IC50 = 1794.2 nM T98711 C4V2RJ 145994271 IC50 = 9880 nM T98711 CC27PZ 146443282 IC50 = 2290 nM T98711 C06YAR 153979960 IC50 = 4000 nM T98711 CJ8V4Q 153979967 IC50 = 600 nM T98711 C5B1RI 153979968 IC50 = 1300 nM T98711 CZ2OW7 153979970 IC50 = 0.07 nM T98711 C2H9LT 153979972 IC50 = 70 nM T98711 CD6EF5 153979973 IC50 = 800 nM T98711 C15LBY 153979974 IC50 > 10000 nM T98711 CTV4G0 153979975 IC50 > 10000 nM T98711 CS4E3M 153979977 IC50 = 0.15 nM T98711 CH6A9F 153979986 IC50 = 9400 nM T98711 CBXN70 153979988 IC50 > 10000 nM T98711 C9L8CY 153979991 IC50 = 80 nM T98711 C94IGO 155510425 IC50 = 301 nM T98711 C0AZ2W 155510575 IC50 = 6030 nM T98711 CRX53K 155510902 IC50 = 426 nM T98711 C2TRD5 155511051 IC50 = 328 nM T98711 CH4PT0 155511056 IC50 > 50000 nM T98711 CQD8U1 155511223 IC50 = 6 nM T98711 C0TY4L 155512256 IC50 > 50000 nM T98711 C30QIL 155512277 IC50 > 50000 nM T98711 CYT0U1 155512533 IC50 = 933.25 nM T98711 CN1L2G 155512563 IC50 = 7060 nM T98711 C2OVJ6 155513058 IC50 > 50000 nM T98711 C8QOL4 155513096 IC50 = 40 nM T98711 CLP7Q5 155513372 IC50 = 2300 nM T98711 C8S4OV 155513382 IC50 > 10000 nM T98711 CQ4MT7 155514267 IC50 > 50000 nM T98711 CE31CI 155514453 IC50 = 2950 nM T98711 CY0E3D 155514519 IC50 = 11000 nM T98711 C4QTY1 155514573 IC50 = 25.6 nM T98711 C36OGK 155514733 IC50 > 50000 nM T98711 CBKQ23 155514904 IC50 = 41.69 nM T98711 CS0C1V 155515351 IC50 = 6.31 nM T98711 C8WO0D 155515901 IC50 = 11700 nM T98711 C37OWC 155516090 IC50 = 13400 nM T98711 CTR7C8 155516568 IC50 = 7220 nM T98711 COIQ70 155516605 IC50 = 67.8 nM T98711 CI02NB 155516607 IC50 = 395 nM T98711 CR4P3Z 155516698 IC50 = 3100 nM T98711 COQ0I2 155517103 IC50 = 8410 nM T98711 C7WQF6 155517133 IC50 = 38.9 nM T98711 C7CN4W 155517273 IC50 = 340 nM T98711 CFG9A1 155517376 IC50 = 54 nM T98711 C0DR8X 155517455 IC50 = 1020 nM T98711 CEU36W 155517463 IC50 > 50000 nM T98711 C62HKG 155518395 IC50 = 206 nM T98711 C0DUP5 155518577 IC50 = 27360 nM T98711 COR6Z3 155518726 IC50 = 65 nM T98711 CWA5P2 155518864 IC50 > 10000 nM T98711 CT5X0O 155519170 IC50 = 12.59 nM T98711 C0XI2C 155519241 IC50 = 48.2 nM T98711 CWOJ19 155519277 IC50 = 2740 nM T98711 CET82F 155519354 IC50 = 5300 nM T98711 CEJ87B 155519446 IC50 = 180 nM T98711 C1DVS3 155519968 IC50 = 125.3 nM T98711 CW65KH 155520207 IC50 = 140 nM T98711 CAIX71 155520508 IC50 > 10000 nM T98711 CZR0D3 155520717 IC50 = 5500 nM T98711 CHG5D0 155521756 IC50 = 7300 nM T98711 C9AT3Q 155521926 IC50 = 0.0017 nM T98711 CC2U3Z 155522419 IC50 = 1210 nM T98711 C2ML7G 155522745 IC50 = 9970 nM T98711 CF1OL6 155523160 IC50 = 4520 nM T98711 C1AEU5 155523624 IC50 = 48.98 nM T98711 C2ES7G 155523649 IC50 = 3900 nM T98711 CU0E6I 155523688 IC50 = 251.19 nM T98711 CS6IJ2 155524198 IC50 > 30000 nM T98711 C9VWZ8 155524523 IC50 = 79.43 nM T98711 CH24YB 155525250 IC50 = 398.11 nM T98711 CGMH43 155525252 IC50 = 64 nM T98711 C32XUD 155525503 IC50 = 190.55 nM T98711 CNB25L 155525773 IC50 > 100000 nM T98711 C3K9OH 155526042 IC50 = 13.18 nM T98711 CMT9X3 155526434 IC50 = 2.512 nM T98711 C6NU8X 155526479 IC50 = 56 nM T98711 CDY49N 155526514 IC50 = 501.19 nM T98711 CK85TG 155526796 IC50 = 123 nM T98711 CU0X9B 155526812 IC50 = 7.413 nM T98711 C9ZR4K 155526939 IC50 = 32.6 nM T98711 C68XKW 155527023 IC50 = 307 nM T98711 C1UOP6 155528201 IC50 = 4520 nM T98711 CR7VW0 155528538 IC50 > 10000 nM T98711 C68UIE 155528833 IC50 > 100000 nM T98711 CE98VB 155529070 IC50 = 2400 nM T98711 CC25TX 155530201 IC50 > 100000 nM T98711 CT80OY 155530802 IC50 = 158.49 nM T98711 C1V6BO 155531034 IC50 = 0.17 nM T98711 C2GH4F 155531521 IC50 = 3100 nM T98711 C3E5FM 155531627 IC50 = 140 nM T98711 CWB5N8 155532073 IC50 = 6420 nM T98711 C15PWD 155532152 IC50 = 36.1 nM T98711 C6XQF3 155532358 IC50 = 174 nM T98711 C3G4ZQ 155532469 IC50 = 970 nM T98711 CE13NX 155532485 IC50 = 32.36 nM T98711 CQL91M 155532503 IC50 = 55 nM T98711 C4I0CS 155533039 IC50 > 50000 nM T98711 CW1X5G 155533337 IC50 = 39000 nM T98711 C2ZAO9 155533687 IC50 = 1737.8 nM T98711 C8Q0OL 155533954 IC50 = 1100 nM T98711 CYN5O8 155534304 IC50 = 740 nM T98711 C9W7XG 155534725 IC50 = 9000 nM T98711 C76NZI 155535091 IC50 = 18000 nM T98711 CLOD29 155535170 IC50 = 500 nM T98711 CMY84N 155535601 IC50 = 27 nM T98711 CS5A6Y 155535996 IC50 = 190 nM T98711 CT90DI 155536211 IC50 = 290 nM T98711 CKI2M0 155536368 IC50 = 398.11 nM T98711 CY4D3B 155537306 IC50 = 520 nM T98711 C6R7XI 155537540 IC50 = 2.92 nM T98711 CB8CJ4 155538052 IC50 = 63 nM T98711 CA6EU8 155538194 IC50 = 15800 nM T98711 CGI1P4 155539252 IC50 = 48.6 nM T98711 C5WI2G 155539893 IC50 > 10000 nM T98711 C9JWY1 155540039 IC50 = 9360 nM T98711 C4RY7K 155540049 IC50 = 55.7 nM T98711 CRW71X 155540051 IC50 = 169 nM T98711 CM3G5X 155540209 IC50 = 7762.47 nM T98711 CVKX83 155540924 IC50 > 10000 nM T98711 CE1UC4 155541278 IC50 > 10000 nM T98711 CMT9Q2 155541386 IC50 = 70.2 nM T98711 CI64ZO 155541480 IC50 > 30000 nM T98711 CJA34X 155541507 IC50 = 48.6 nM T98711 C2PA7S 155542132 IC50 = 9.9 nM T98711 C8CM4P 155542748 IC50 = 120 nM T98711 C9KR0B 155542856 IC50 = 5310 nM T98711 CMO67L 155543176 IC50 = 568 nM T98711 CSKI49 155543595 IC50 = 86.1 nM T98711 C0RFH7 155543896 IC50 = 11.48 nM T98711 C17JEA 155543947 IC50 = 300 nM T98711 CH7ZX3 155544057 IC50 = 92.6 nM T98711 CV4MO2 155544490 IC50 = 4600 nM T98711 CNQ0F4 155544914 IC50 = 6070 nM T98711 C3FTK8 155545055 IC50 > 50000 nM T98711 CMXY60 155545085 IC50 > 10000 nM T98711 C7NA0J 155545226 IC50 = 135000 nM T98711 C79JFO 155545405 IC50 = 4520 nM T98711 C6C7AM 155545895 IC50 = 123.03 nM T98711 COW1Z3 155546180 IC50 = 6.06 nM T98711 CM6QN1 155546316 IC50 = 390 nM T98711 C35VQY 155546517 IC50 = 4520 nM T98711 C9WA1M 155546797 IC50 > 50000 nM T98711 CBPS95 155546845 IC50 > 10000 nM T98711 CPYV79 155547224 IC50 > 50000 nM T98711 CD9I8N 155547289 IC50 = 55.9 nM T98711 CX32QR 155547425 IC50 = 6.5 nM T98711 CS60BV 155547778 IC50 = 74.8 nM T98711 C4TQ5J 155548079 IC50 = 21.1 nM T98711 C5VMU7 155548207 IC50 = 21.8 nM T98711 CD8JZ5 155548223 IC50 > 30000 nM T98711 C4Q7RL 155548245 IC50 = 41.5 nM T98711 CK8RB0 155548367 IC50 = 5890000 nM T98711 C91ODF 155548523 IC50 = 910 nM T98711 CP85KA 155548858 IC50 = 480 nM T98711 CDEL58 155549426 IC50 = 26.7 nM T98711 CFT71V 155549427 IC50 = 199 nM T98711 CA8FQ3 155549571 IC50 = 1090 nM T98711 C5UC0N 155549656 IC50 = 29000 nM T98711 C94KDL 155550161 IC50 = 3.9 nM T98711 C0A7KH 155550386 IC50 = 8690 nM T98711 C2DYJ7 155551094 IC50 = 17.5 nM T98711 CAY6R5 155551298 IC50 = 27000 nM T98711 CUCF03 155551499 IC50 = 140 nM T98711 C31YDU 155551611 IC50 > 50000 nM T98711 CM2X5O 155551629 IC50 = 110 nM T98711 C5U0SM 155552824 IC50 = 93.7 nM T98711 CJXS06 155552844 IC50 = 251.19 nM T98711 CD87VC 155553046 IC50 = 0.497 nM T98711 CQ2SG6 155554219 IC50 = 6900 nM T98711 CRZW49 155554295 IC50 > 50000 nM T98711 C0P6IW 155554556 IC50 = 196 nM T98711 CS54UQ 155554734 IC50 = 1910 nM T98711 C0W3LZ 155554767 IC50 = 120 nM T98711 CFNH83 155554841 IC50 = 304 nM T98711 C8Z0MS 155555442 IC50 > 50000 nM T98711 CFK23R 155555484 IC50 = 83.7 nM T98711 C7N1YW 155555576 IC50 = 68.2 nM T98711 C53TJU 155555938 IC50 = 1148.15 nM T98711 CCHJ45 155555939 IC50 = 80.6 nM T98711 CHC64Z 155556086 IC50 = 219000 nM T98711 CD21TM 155556234 IC50 > 50000 nM T98711 C9YCT8 155556531 IC50 = 0.515 nM T98711 CD5L2W 155556671 IC50 = 9450 nM T98711 C0WAR6 155556705 IC50 = 52 nM T98711 C2EA7Q 155556733 IC50 = 1800 nM T98711 C7S5JN 155556840 IC50 = 19000 nM T98711 CDN6B5 155556926 IC50 = 9.1 nM T98711 C7IRE9 155557054 IC50 = 722 nM T98711 CU1G2L 155557132 IC50 = 1258.93 nM T98711 CK5Q9E 155557224 IC50 = 23 nM T98711 CI41HC 155557480 IC50 = 79.43 nM T98711 CVH23J 155557537 IC50 = 200 nM T98711 CVF40Y 155557821 IC50 = 25 nM T98711 CS28NH 155557943 IC50 = 13 nM T98711 CAMC16 155558019 IC50 = 50.12 nM T98711 CYP20F 155558662 IC50 > 50000 nM T98711 CE8PZ1 155559190 IC50 = 11000 nM T98711 C82GCI 155559240 IC50 = 74 nM T98711 C4T7HU 155560397 IC50 = 232 nM T98711 C0SQ7I 155560420 IC50 = 5800 nM T98711 CI8UF7 155560617 IC50 > 30000 nM T98711 C2VCE7 155560793 IC50 = 8250 nM T98711 CLY7Q6 155560920 IC50 > 30000 nM T98711 CHSY32 155560934 IC50 = 19.8 nM T98711 C95CBX 155561050 IC50 = 3900 nM T98711 CP7I9L 155561118 IC50 > 30000 nM T98711 C15FIN 155561744 IC50 = 630.96 nM T98711 CR12EX 155561772 IC50 = 4710 nM T98711 C0A9HJ 155562003 IC50 = 185 nM T98711 CCUM34 155562078 IC50 > 50000 nM T98711 CUZ64A 155562266 IC50 = 130 nM T98711 C7USO2 155562419 IC50 = 4520 nM T98711 C92PGF 155563169 IC50 = 3540 nM T98711 CJQ59S 155563181 IC50 = 7830 nM T98711 CU6NW2 155563256 IC50 = 22.9 nM T98711 CAP30C 155563421 IC50 = 4650 nM T98711 CTK04N 155563892 IC50 > 10000 nM T98711 C5HT8V 155564601 IC50 > 100000 nM T98711 CY6OR7 155564797 IC50 = 800 nM T98711 C27WPT 155565176 IC50 = 748 nM T98711 C5OTD7 155566135 IC50 = 34.67 nM T98711 C7NJY2 155566392 IC50 = 3500 nM T98711 C2NB9W 155566555 IC50 = 14000 nM T98711 CWPL14 155566983 IC50 = 68000 nM T98711 C9R2MS 155567099 IC50 = 78 nM T98711 CNQ18H 155567205 IC50 = 6.95 nM T98711 CM63EC 155567324 IC50 = 39.81 nM T98711 C40XPW 155567716 IC50 = 29000 nM T98711 CW3Q7C 155567905 IC50 = 22 nM T98711 C3EPS6 155567920 IC50 = 35.6 nM T98711 CG3BR0 155567943 IC50 > 100000 nM T98711 CRMO93 155567970 IC50 = 7.8 nM T98711 CR24FZ 155568280 IC50 = 600 nM T98711 CJLF85 155568310 IC50 > 50000 nM T98711 CF1J8X 155568638 IC50 > 50000 nM T98711 CDQ05E 155568688 IC50 = 20 nM T98711 C10CZA 155569041 IC50 = 75.7 nM T98711 CZGB74 155569334 IC50 = 65.7 nM T98711 C1YG5A 10015862 IC50 = 138 nM T98711 CB49KJ 10906319 IC50 = 23780 nM T98711 D00AHD 44435223 Ki = 3.5 nM T98711 D00ANJ 1897797 Ki > 100000 nM T98711 D00DKI 10107976 IC50 = 153 nM T98711 D00KTT 44568318 Ki = 18100 nM T98711 D00MFR 44419695 IC50 = 1099.01 nM T98711 D00PLH 44428832 Ki > 100000 nM T98711 D00QLR 10403152 IC50 = 1370 nM T98711 D00RIX 5280443 Ki = 37400 nM T98711 D00VXE 3253193 Ki = 350 nM T98711 D00XHC 12851057 Ki = 180 nM T98711 D01AJQ 46232725 IC50 = 400 nM T98711 D01EZC 44421938 IC50 = 2650 nM T98711 D01FNH 24905597 Ki = 2260 nM T98711 D01HRG 12884 Ki = 68800 nM T98711 D01HZN 44428835 Ki > 100000 nM T98711 D01LVY 3473393 Ki = 2500 nM T98711 D01MAC 25133941 IC50 = 894 nM T98711 D01OND 46080 IC50 = 18000 nM T98711 D01QRR 25130201 IC50 = 6 nM T98711 D01VAU 123493 Ki > 100000 nM T98711 D01VCS 44428837 Ki > 100000 nM T98711 D01XGP 123358 Ki = 2630 nM T98711 D01XKY 3473392 Ki = 1300 nM T98711 D02BDL 8433 Ki > 100000 nM T98711 D02DUJ 65719 IC50 = 12 nM T98711 D02GJG 11043027 Ki > 100000 nM T98711 D02HQS 19377173 Ki > 100000 nM T98711 D02LWX 44419700 IC50 = 8700 nM T98711 D02SGJ 19009 IC50 > 100000 nM T98711 D02TLP 11363 Ki > 100000 nM T98711 D02XHM 44421959 IC50 = 100 nM T98711 D02YSX 197033 IC50 = 7900000 nM T98711 D03HZT 89076 Ki > 100000 nM T98711 D03NTO 25129142 IC50 = 57 nM T98711 D03OGO 465614 IC50 = 770 nM T98711 D03TPH 87203 Ki > 100000 nM T98711 D04AWS 704267 Ki = 2990 nM T98711 D04AXR 96047 Ki > 100000 nM T98711 D04CDV 44428829 Ki > 100000 nM T98711 D04CTO 44435201 Ki = 1700 nM T98711 D04EXR 251908 Ki > 100000 nM T98711 D04FHZ 9906452 IC50 = 1950 nM T98711 D04GTP 23645738 IC50 = 1700 nM T98711 D04IXN 16645663 Ki = 10500 nM T98711 D04JCW 25128787 IC50 = 700 nM T98711 D04PKD 25129847 IC50 = 980 nM T98711 D04SYM 25129843 IC50 = 5100 nM T98711 D04ZWS 11173982 IC50 = 260 nM T98711 D04ZZU 24905653 Ki = 570 nM T98711 D05AVX 60983 Ki > 100000 nM T98711 D05DIN 24905595 Ki = 340 nM T98711 D05EMT 22574258 Ki > 100000 nM T98711 D05EYA 18946 Ki > 100000 nM T98711 D05GPI 44421960 IC50 = 120 nM T98711 D05LTW 22574224 Ki = 1270 nM T98711 D05PNO 4135273 Ki > 100000 nM T98711 D05QFR 25133942 IC50 = 2500 nM T98711 D05UJV 52945624 IC50 = 16000 nM T98711 D05VLV 3473842 Ki = 1900 nM T98711 D05VUC 19971657 Ki > 100000 nM T98711 D05XPW 46232686 IC50 = 1220 nM T98711 D05XRY 2752926 Ki > 100000 nM T98711 D05ZCX 44435802 Ki > 100000 nM T98711 D06BDB 25128786 IC50 = 4100 nM T98711 D06ERH 637760 IC50 = 87000 nM T98711 D06FFD 96430 Ki > 100000 nM T98711 D06GYH 16745302 Ki > 100000 nM T98711 D06KQH 10178151 IC50 = 1580 nM T98711 D06UXW 107759 IC50 = 977.24 nM T98711 D06VGD 6724 Ki = 2970 nM T98711 D06YEB 44435197 Ki = 1700 nM T98711 D06ZRX 5281717 IC50 = 2950 nM T98711 D07AYF 3107576 Ki = 10200 nM T98711 D07CFJ 589576 Ki > 100000 nM T98711 D07EDG 1901244 Ki = 12600 nM T98711 D07RIQ 71028 IC50 > 10000 nM T98711 D07YJG 11351920 IC50 = 7000 nM T98711 D08AOG 90571 Ki > 100000 nM T98711 D08BKE 44568822 IC50 = 359 nM T98711 D08FQW 24905593 Ki = 1690 nM T98711 D08NNF 46229054 Ki = 10000 nM T98711 D08PWL 52945680 IC50 = 70000 nM T98711 D08TBI 24905535 Ki = 3190 nM T98711 D08UET 4939 IC50 = 13200 nM T98711 D08UOB 44428840 Ki > 100000 nM T98711 D08XQI 9395 IC50 = 7 nM T98711 D08ZLS 705757 Ki = 4450 nM T98711 D09ALJ 5280805 Ki = 501200 nM T98711 D09CGV 44419702 IC50 = 1625.55 nM T98711 D09DWA 3473839 Ki = 3100 nM T98711 D09GKY 705769 Ki = 2810 nM T98711 D09GXM 44421953 IC50 = 800 nM T98711 D09HZE 705776 Ki = 7100 nM T98711 D09LSR 11437501 Ki > 100000 nM T98711 D09OPL 705775 Ki = 1560 nM T98711 D09QDC 5420 IC50 = 733 nM T98711 D09YLY 25129143 IC50 = 88 nM T98711 D0A0YX 5143 IC50 = 3600 nM T98711 D0A5FO 222149 Ki = 220 nM T98711 D0AQ3K 44421955 IC50 = 100 nM T98711 D0AW4P 10868634 Ki > 100000 nM T98711 D0B0ZM 2235291 Ki = 430 nM T98711 D0B1TQ 1810509 Ki > 100000 nM T98711 D0B4DT 44421954 IC50 = 80 nM T98711 D0B6IQ 2301676 Ki = 9200 nM T98711 D0B8YX 75511 Ki > 100000 nM T98711 D0BB2U 2385968 Ki > 100000 nM T98711 D0C0XU 10496398 IC50 = 40 nM T98711 D0C1LI 53378764 IC50 = 1820 nM T98711 D0C9AD 277990 Ki = 21900 nM T98711 D0CN8Z 11392969 Ki > 100000 nM T98711 D0D0BI 8371 Ki = 268 nM T98711 D0D2HH 44428834 Ki > 100000 nM T98711 D0D7FN 283893 Ki > 100000 nM T98711 D0D7MN 44435217 Ki = 88 nM T98711 D0D8IH 777336 Ki = 310 nM T98711 D0DB9T 704261 Ki = 10600 nM T98711 D0DR7A 934131 Ki = 12100 nM T98711 D0DV9Z 44419694 IC50 = 20900 nM T98711 D0DW9J 123072 Ki > 100000 nM T98711 D0E2IG 44428839 Ki > 100000 nM T98711 D0E4GM 16728608 IC50 = 3600 nM T98711 D0E5ZP 604575 Ki > 100000 nM T98711 D0EI5V 16115140 IC50 = 40000 nM T98711 D0EK7H 2734793 Ki > 100000 nM T98711 D0EQ1Z 45487256 IC50 = 1.2 nM T98711 D0ER5C 44419701 IC50 = 32200 nM T98711 D0F3QP 5889042 IC50 = 2570 nM T98711 D0F3RN 89801 Ki > 100000 nM T98711 D0F5EJ 11375002 IC50 = 10.8 nM T98711 D0F5VY 94860 Ki = 1670 nM T98711 D0FO2B 1923 IC50 > 100 nM T98711 D0FP5F 46232685 IC50 = 10400 nM T98711 D0G0ED 44420671 IC50 = 790 nM T98711 D0G0GZ 19916609 Ki = 18300 nM T98711 D0G2DQ 4669250 Ki > 100000 nM T98711 D0G2WI 10318177 IC50 = 4500 nM T98711 D0G3TK 5280863 Ki = 43100 nM T98711 D0G5TL 44419706 IC50 = 2685.34 nM T98711 D0H1NU 10135721 IC50 = 3520 nM T98711 D0H2UG 52946279 IC50 = 360 nM T98711 D0H3BC 44421943 IC50 = 2490 nM T98711 D0H3WJ 44435193 Ki = 560 nM T98711 D0I3XA 6422124 IC50 = 77300 nM T98711 D0I4LX 1403 IC50 = 3370 nM T98711 D0I5LV 24905596 Ki = 710 nM T98711 D0I7BX 16645664 Ki = 36 nM T98711 D0IC5U 11573367 IC50 = 3.6 nM T98711 D0J1IX 1238015 Ki = 610 nM T98711 D0J3SN 1868 IC50 > 10000 nM T98711 D0J5AU 25133940 IC50 = 3900 nM T98711 D0J8LQ 607810 Ki = 600 nM T98711 D0JH7C 72810 Ki > 100000 nM T98711 D0JI0H 3542734 Ki = 28100 nM T98711 D0K3YM 704259 Ki = 3410 nM T98711 D0K6OM 44428838 Ki > 100000 nM T98711 D0K6PO 316765 Ki > 100000 nM T98711 D0K7EC 705771 Ki = 1050 nM T98711 D0K8BT 25129490 IC50 = 669 nM T98711 D0L1EI 9969234 IC50 = 1890 nM T98711 D0L1ST 2777298 Ki > 100000 nM T98711 D0L3EE 262319 Ki = 5800 nM T98711 D0L4MF 44428833 Ki > 100000 nM T98711 D0L4OW 9823294 IC50 = 310 nM T98711 D0L5QJ 11408144 IC50 = 6000 nM T98711 D0L9YJ 44421937 IC50 = 8330 nM T98711 D0LJ2F 11806279 Ki > 100000 nM T98711 D0LL8H 25129141 IC50 = 4.3 nM T98711 D0M0BM 10399068 IC50 = 114 nM T98711 D0M2EM 4650 Ki = 2050 nM T98711 D0M2LD 1476756 IC50 > 1000000 nM T98711 D0M2TY 10168 IC50 = 17000 nM T98711 D0M2ZD 44428831 Ki > 100000 nM T98711 D0M4IE 9549196 Ki = 0.163 nM T98711 D0M5NR 3794313 Ki > 100000 nM T98711 D0M6IJ 44435218 Ki = 470 nM T98711 D0MF5Y 5281614 Ki = 90000 nM T98711 D0N0HK 73252 Ki = 3200 nM T98711 D0N6XS 44435196 Ki = 400 nM T98711 D0N8YZ 2427416 Ki > 100000 nM T98711 D0N9ZR 1718647 Ki = 56500 nM T98711 D0NJ4G 80771 Ki > 100000 nM T98711 D0NJ5W 10055202 IC50 = 11600 nM T98711 D0O0LU 264734 Ki > 100000 nM T98711 D0O2OH 9907847 IC50 = 50 nM T98711 D0O8DZ 44421948 IC50 = 1430 nM T98711 D0O8LK 16066832 IC50 = 150 nM T98711 D0O9YQ 52941983 IC50 = 1000 nM T98711 D0OJ9P 49799304 IC50 = 550 nM T98711 D0P1IK 44428841 Ki > 100000 nM T98711 D0P3VH 893336 Ki = 6200 nM T98711 D0P7TN 465615 IC50 = 4600 nM T98711 D0PF7F 9928397 IC50 = 1950 nM T98711 D0PQ5R 24905594 Ki = 2850 nM T98711 D0Q0BV 24905710 Ki = 120 nM T98711 D0Q2YJ 6763 Ki = 190 nM T98711 D0Q3EV 52948017 IC50 = 120 nM T98711 D0R2GR 46229025 Ki = 2660 nM T98711 D0R2QC 10275242 IC50 = 31550 nM T98711 D0S1MC 23643351 IC50 = 118000 nM T98711 D0S2DW 9844749 IC50 = 48900 nM T98711 D0S3WF 10222714 IC50 = 1350 nM T98711 D0S6TW 1845 Ki > 100000 nM T98711 D0S8AS 44568319 Ki = 4300 nM T98711 D0S9YA 638276 IC50 = 84000 nM T98711 D0SP2O 7054 Ki > 100000 nM T98711 D0T3PW 5281672 Ki = 71000 nM T98711 D0T5MD 25128788 IC50 = 334 nM T98711 D0T5XC 31494 Ki > 100000 nM T98711 D0U0BV 44428830 Ki > 100000 nM T98711 D0U3JD 16358 Ki > 100000 nM T98711 D0U7BQ 24905592 Ki = 390 nM T98711 D0U9AU 11385845 IC50 = 6 nM T98711 D0UK5A 76996 Ki > 100000 nM T98711 D0UT1X 101375 Ki > 100000 nM T98711 D0UZ8R 71043 Ki > 100000 nM T98711 D0V4RD 3112604 Ki = 820 nM T98711 D0V7EK 3773589 Ki = 570 nM T98711 D0V8PE 24905534 Ki = 13400 nM T98711 D0W4WB 25129492 IC50 = 3700 nM T98711 D0W9VA 10667 Ki = 2290 nM T98711 D0WB1D 10221700 IC50 = 560 nM T98711 D0WH4J 25129844 IC50 = 639 nM T98711 D0WX6R 3477013 Ki = 3100 nM T98711 D0X0ER 344135 Ki = 30600 nM T98711 D0X4HG 10765787 IC50 = 48 nM T98711 D0X7CW 497286 IC50 = 350 nM T98711 D0XI4U 5319470 IC50 = 17458.22 nM T98711 D0XL1R 9976105 IC50 = 2915 nM T98711 D0Y0UV 19916610 Ki = 710 nM T98711 D0Y0XQ 2779383 Ki > 100000 nM T98711 D0Y2TE 10112356 IC50 = 5230 nM T98711 D0Y5KN 44568823 IC50 = 72 nM T98711 D0Y6RZ 22574214 Ki > 100000 nM T98711 D0Y7FX 8651 Ki > 100000 nM T98711 D0Y7HG 5281616 Ki = 6900 nM T98711 D0YZ3E 44435200 Ki = 220 nM T98711 D0Z1WQ 76915 Ki > 100000 nM T98711 D0Z5KQ 8400 Ki > 100000 nM T98711 D0Z6CZ 5139980 Ki > 100000 nM T98711 D0Z6DK 44423026 IC50 > 50000 nM T98711 D0Z6WU 201563 IC50 = 5000 nM T98711 D0Z8HX 16786802 Ki > 100000 nM T98711 D0ZI7F 211174 IC50 = 17400 nM T98711 D0ZL6B 3772674 Ki > 100000 nM T98711 D0ZR2T 2732752 Ki > 100000 nM T98711 D0ZT5C 44428828 Ki > 100000 nM T61729 CMO39B 7493 Ki = 2600 nM T61729 C4VE6C 192744 Ki = 140 nM T61729 C19UCJ 60018837 Ki = 200 nM T47941 D05MQK 110635 IC50 = 9200 nM T47941 D07ESC 11561674 IC50 = 74 nM T47941 D09AMZ 1676 Ki = 43100 nM T47941 D09QEI 4740 Ki = 37700 nM T47941 D0C9SY 135400189 IC50 = 3800 nM T47941 D0E0SW 53708 IC50 = 2900 nM T47941 D0F8RA 2153 Ki = 56800 nM T47941 D0F9GE 3108 IC50 = 500 nM T47941 D0R4UW 449193 IC50 = 0.8 nM T47941 D0U7GK 5426 IC50 > 500000 nM T47941 D0Y9ZE 4197 IC50 = 6000 nM T47941 D0Z7ZM 135398744 IC50 > 500 nM T47941 D01XHG 2984 IC50 = 170 nM T47941 D0DK8X 50922691 IC50 = 5600 nM T47941 D0F4TV 6918428 IC50 = 14 nM T47941 D0M3IN 1188 Ki > 200000 nM T47941 D0M5BS 9864321 IC50 = 0.08 nM T47941 D0M7CB 9919680 IC50 = 5.1 nM T47941 D0SM0W 44591583 IC50 = 110 nM T47941 D0T5PO 5092 Ki = 1.6 nM T47941 D0U2DH 9844338 IC50 = 1100 nM T47941 D0X0PP 59351313 IC50 > 30000 nM T47941 D0Z2FB 154575 Ki = 0.4 nM T47941 D0LF0O 135441202 IC50 = 4000 nM T47941 D07EUB 46200734 IC50 = 4820 nM T47941 D00DBE 9865514 IC50 = 1100 nM T47941 D00SPK 23665864 IC50 = 3400 nM T47941 D00YPW 135399235 IC50 = 53000 nM T47941 D01FRF 5537 IC50 = 400 nM T47941 D01FXD 9802841 IC50 = 60 nM T47941 D01QUF 9842576 Ki = 1 nM T47941 D02EMR 151170 IC50 = 10 nM T47941 D07FHZ 5087 IC50 = 4800 nM T47941 D08SNX 135430158 Ki = 436 nM T47941 D09UMA 55918 IC50 = 6000 nM T47941 D0E9PT 127769 IC50 = 2000 nM T47941 D0F0CS 5723 IC50 = 158.49 nM T47941 D0K2BQ 71356 IC50 = 1900 nM T47941 D0SI4C 126487 IC50 = 12000 nM T47941 D0UG4T 127928 IC50 = 4.5 nM T47941 CO2Y3R 3698 IC50 = 41000 nM T47941 C3B8VG 5369 IC50 = 4700 nM T47941 C0QUJ8 23102 IC50 = 1640 nM T47941 C1TI6Y 32014 IC50 = 7700 nM T47941 CY8K9D 70639 Ki = 156000 nM T47941 C6N3XY 91636 IC50 = 200000 nM T47941 C8RE9U 94432 IC50 = 17000 nM T47941 CW0S8Y 100299 IC50 = 22000 nM T47941 C8HDQ3 121397 IC50 > 1000000 nM T47941 CZ39NL 127770 IC50 = 37000 nM T47941 CGA17S 127779 Ki = 2000 nM T47941 CS7AB0 130604 IC50 = 16 nM T47941 C5N6TM 161713 Ki = 28600 nM T47941 CVQ8D3 169185 IC50 = 33000 nM T47941 CEG2T8 169316 Ki = 10200 nM T47941 CN1V0P 174907 Ki = 26000 nM T47941 C03NBI 192356 IC50 = 740 nM T47941 C0Y8GT 218667 Ki = 32000 nM T47941 C8FWD2 317789 IC50 = 1258.93 nM T47941 C7QO3K 343627 Ki = 32400 nM T47941 C8EFH4 349956 IC50 = 1800 nM T47941 C9GV7U 350737 Ki = 63000 nM T47941 C89XKO 367855 IC50 = 6000 nM T47941 C7FU6V 403193 IC50 = 3700 nM T47941 C2EF5G 404497 IC50 = 1300 nM T47941 CPE2J7 461663 IC50 = 9400 nM T47941 CNH7C2 461664 IC50 = 2500 nM T47941 C8TI2H 464987 IC50 = 4700 nM T47941 C6SQ2O 551348 IC50 = 19000 nM T47941 C63NXL 557364 IC50 = 9000 nM T47941 CC5L4Y 557426 IC50 = 1100 nM T47941 CT1D5G 566496 IC50 = 1020 nM T47941 C8V2BG 583390 IC50 = 6000 nM T47941 CV6ZB1 608456 IC50 = 50000 nM T47941 C95VXQ 659516 Ki > 100000 nM T47941 CDV1A0 662394 IC50 = 12600000 nM T47941 CQU82Z 662872 IC50 = 8400000 nM T47941 C1B6ZL 662965 IC50 = 40000 nM T47941 C4N1QH 667701 IC50 = 4300 nM T47941 CVHU85 694543 IC50 = 20000 nM T47941 CX4PH9 935803 IC50 = 12500000 nM T47941 C8EYM9 1499306 IC50 = 88900 nM T47941 CSL45P 2380588 IC50 = 1584.89 nM T47941 C4KQ7E 2800759 IC50 = 10000 nM T47941 C5D6NL 2822835 IC50 = 1500 nM T47941 C3P0TU 2822850 IC50 = 6400 nM T47941 CAQV87 2822851 IC50 = 9 nM T47941 CNO2S1 2822853 IC50 = 4100 nM T47941 CS3Y1H 2822859 IC50 = 6550 nM T47941 CML54G 2822864 IC50 = 10000 nM T47941 CFB78N 2822879 IC50 = 56000 nM T47941 CA7F9Y 2822887 IC50 = 320 nM T47941 C5JF8U 2822888 IC50 = 6010 nM T47941 C37MVS 2823055 IC50 = 80 nM T47941 C61NHX 2823068 IC50 = 670 nM T47941 CFI1M9 3010411 IC50 = 60000 nM T47941 CW4HY0 3024653 IC50 = 1200 nM T47941 C94YRH 3024655 IC50 = 300 nM T47941 CD81TE 3071939 IC50 = 2000 nM T47941 CK69NE 3071940 IC50 = 2500 nM T47941 CQXU38 3071959 IC50 = 6600 nM T47941 C1TSP2 3071969 IC50 = 520 nM T47941 C3XHS9 3071971 IC50 = 150 nM T47941 CS3G6W 3071975 IC50 = 3600 nM T47941 CB42XD 3073378 IC50 = 140 nM T47941 C5RWI8 3244396 IC50 = 14100000 nM T47941 CN98CX 3393127 IC50 = 6300000 nM T47941 CU91IC 3435529 IC50 = 126000 nM T47941 CW2X0T 3492181 IC50 = 177000 nM T47941 CG8RD0 3636010 Ki = 36500 nM T47941 COP24T 3788138 IC50 = 7500000 nM T47941 CJ2X5E 3829988 IC50 = 141000 nM T47941 CT56DJ 3835979 IC50 = 10100000 nM T47941 C8JZ9N 3849553 IC50 = 8900000 nM T47941 CX1H6T 4363048 IC50 = 12600000 nM T47941 C91CHU 4558271 IC50 = 8400000 nM T47941 CBS67I 5271722 IC50 = 11000 nM T47941 CR5GH1 5284402 Ki = 5.4 nM T47941 CFES14 5311486 IC50 = 5700 nM T47941 CV1ZT5 5332193 IC50 > 10000 nM T47941 CEQO37 5332328 IC50 = 4900 nM T47941 CM47KI 5351344 IC50 > 10000 nM T47941 CL3DY5 5487421 IC50 = 118000 nM T47941 CUH3P2 5488456 IC50 = 348000 nM T47941 C6W1VO 5939551 IC50 = 8200 nM T47941 C83NVB 6109780 IC50 > 10000 nM T47941 CAYS61 6918354 IC50 = 0.63 nM T47941 CB40PM 6918356 IC50 = 0.13 nM T47941 CR0NJ7 6918510 IC50 = 30000 nM T47941 C1XP7Q 7659902 IC50 = 60 nM T47941 CJO4P1 9580443 IC50 = 10000 nM T47941 CNC2F4 9798336 IC50 = 66 nM T47941 CB3L7K 9799054 IC50 = 6.8 nM T47941 CFJ62Y 9799389 IC50 = 67.6 nM T47941 C3EOU7 9799418 IC50 = 39.81 nM T47941 C8QEW1 9800492 IC50 = 1500 nM T47941 CFRM61 9800710 Ki = 473 nM T47941 C0SGZ3 9801104 IC50 = 21 nM T47941 CET56A 9801414 IC50 = 30 nM T47941 CDZP94 9801613 IC50 = 340 nM T47941 C87ERL 9806003 IC50 = 7.943 nM T47941 CHK3Z5 9806981 IC50 = 3.981 nM T47941 CWGO48 9808563 IC50 = 5.012 nM T47941 C7NR8P 9814956 IC50 > 100 nM T47941 CXF0J7 9818343 IC50 = 4800 nM T47941 C1CXA5 9818702 IC50 = 40 nM T47941 C3F1RK 9818713 IC50 = 150 nM T47941 C7YI2H 9821148 IC50 = 1 nM T47941 C4NHZ3 9821373 IC50 = 220 nM T47941 CMUD24 9822422 IC50 = 14 nM T47941 CGH2J9 9822515 IC50 = 410 nM T47941 CDU8L4 9824184 IC50 = 690 nM T47941 C36BNO 9824509 IC50 = 38.9 nM T47941 C0K3SA 9825739 IC50 = 700 nM T47941 C7B1PO 9826435 IC50 = 40 nM T47941 C3OCG4 9826530 Ki = 13 nM T47941 CKG34S 9828282 IC50 = 15.85 nM T47941 CKOT49 9829555 IC50 = 6.31 nM T47941 C56QMD 9836656 IC50 > 100 nM T47941 CK7E8D 9839760 IC50 = 1640 nM T47941 CL70YN 9840066 IC50 = 24 nM T47941 C28YZC 9841233 IC50 = 170 nM T47941 CEW4G2 9842857 IC50 = 195 nM T47941 CUMK40 9843423 IC50 = 149.97 nM T47941 CYI10W 9843466 IC50 = 25 nM T47941 C2FHQ6 9843774 IC50 = 239.88 nM T47941 C4RB2T 9844893 IC50 = 144.54 nM T47941 CAI32D 9844913 IC50 = 120 nM T47941 C6TD8Z 9844923 IC50 = 3.2 nM T47941 CBF06T 9846249 IC50 = 260 nM T47941 CW9D7B 9846655 Ki = 16 nM T47941 CE9F8G 9850007 IC50 = 6 nM T47941 C3ZNU4 9850384 IC50 = 1.995 nM T47941 CFV1Q4 9852021 IC50 = 0.1995 nM T47941 C8QJ4D 9859958 IC50 = 1400 nM T47941 C4F9DV 9861562 IC50 = 340 nM T47941 CN3T1P 9861604 IC50 = 44 nM T47941 C5S0XN 9863370 IC50 = 70 nM T47941 CJ58AE 9864542 IC50 = 28.18 nM T47941 CLF52J 9865916 IC50 = 52.48 nM T47941 C5BQJ8 9865957 IC50 = 4900 nM T47941 CR01PJ 9865970 IC50 = 59 nM T47941 C3HJB5 9867688 IC50 = 1.259 nM T47941 CDW03H 9867844 IC50 = 63.1 nM T47941 CEI5P4 9868140 IC50 = 3000 nM T47941 CVP6S0 9869611 IC50 = 100 nM T47941 CAY84B 9869820 IC50 = 75 nM T47941 CF18MC 9874535 IC50 = 3300 nM T47941 C09UTO 9880681 IC50 > 100 nM T47941 C7XYK6 9881656 IC50 = 1600 nM T47941 C95AMZ 9882035 IC50 = 600 nM T47941 CQJ71T 9887909 IC50 = 3.981 nM T47941 CY65BZ 9894329 IC50 = 2.512 nM T47941 CD6IG8 9894586 IC50 = 30000 nM T47941 CZLA09 9903789 IC50 = 1900 nM T47941 COFA38 9905352 IC50 = 310 nM T47941 CET1I4 9906369 IC50 = 400 nM T47941 C24KBP 9909217 IC50 = 131.83 nM T47941 CW58HA 9910644 IC50 = 75 nM T47941 CWK07N 9911083 IC50 = 12 nM T47941 CISV15 9912092 IC50 = 610 nM T47941 CMBO89 9912467 IC50 = 2.8 nM T47941 C1UL3W 9924218 IC50 > 100 nM T47941 C76RTB 9924539 IC50 = 126 nM T47941 C5MIR1 9926500 IC50 = 1200 nM T47941 CC5K1L 9928654 IC50 = 33 nM T47941 CVNQ72 9930237 IC50 = 59 nM T47941 C2DU3Z 9931012 IC50 = 220 nM T47941 C8JF0Q 9931477 IC50 = 65 nM T47941 CG5AD0 9931784 IC50 = 1.3 nM T47941 CS21YP 9945538 IC50 = 0.52 nM T47941 C81XNB 9949129 IC50 = 440 nM T47941 CB17HL 9949622 IC50 = 1300 nM T47941 C0XTQ5 9950240 IC50 = 230 nM T47941 C9Z8CD 9951712 IC50 = 7.943 nM T47941 CWY06V 9951791 IC50 = 72 nM T47941 CC7R2K 9952592 IC50 = 37 nM T47941 C2CT1U 9955212 IC50 = 120 nM T47941 COS23J 9956462 IC50 = 3.981 nM T47941 C8M2RB 9956613 IC50 = 6.9 nM T47941 C19FKZ 9958988 IC50 = 2.512 nM T47941 C4P8WX 9959207 IC50 = 15.85 nM T47941 C74GQW 9960211 IC50 = 1.4 nM T47941 C2ETO7 9966486 IC50 = 5 nM T47941 CY67GX 9969512 IC50 > 300 nM T47941 CUSE46 9970773 Ki = 32800 nM T47941 CY1J2U 9970847 Ki = 92000 nM T47941 C5W7SI 9970995 IC50 = 1584.89 nM T47941 CN3F0H 9971635 Ki > 200000 nM T47941 CWPA26 9978586 IC50 = 4.1 nM T47941 CQ40MX 9981320 IC50 = 3800 nM T47941 CCXH62 9982563 IC50 = 0.58 nM T47941 C20XIY 9985391 IC50 = 1500 nM T47941 C3G5ZH 9993017 Ki = 56300 nM T47941 C5MX0B 9994095 Ki = 40 nM T47941 CV6TO1 9995407 IC50 = 249 nM T47941 CA9YF5 9998837 IC50 = 851 nM T47941 CFPR64 9999276 IC50 = 0.6 nM T47941 C53HZC 9999401 IC50 = 769 nM T47941 CZ6LM7 10000440 IC50 = 165 nM T47941 CH3PB8 10001036 IC50 = 569 nM T47941 C7OKQ5 10002457 IC50 = 10 nM T47941 CYS20P 10004422 IC50 = 9700 nM T47941 C5HC3V 10004686 IC50 = 4.6 nM T47941 C3BFQ0 10014991 Ki = 46400 nM T47941 C3FT9U 10015082 Ki = 28700 nM T47941 CWV14G 10019207 IC50 = 730 nM T47941 CJI4R6 10021978 IC50 = 2.5 nM T47941 C3A6RV 10027487 IC50 = 160 nM T47941 CIQ0L4 10027501 IC50 = 220 nM T47941 C63YOW 10028092 IC50 = 0.52 nM T47941 C1G5XC 10032458 IC50 = 42000 nM T47941 C7SA9X 10037104 Ki = 19400 nM T47941 CUYW65 10039809 IC50 = 17000 nM T47941 CK5VB0 10041530 IC50 = 14000 nM T47941 CGXS34 10043016 IC50 = 900 nM T47941 CCR2P9 10047419 IC50 = 400 nM T47941 C1L2VF 10050865 IC50 = 17 nM T47941 CFG61D 10060524 Ki = 40800 nM T47941 CO2DF3 10061430 Ki = 60000 nM T47941 C83KZS 10061449 Ki = 26200 nM T47941 C1W2BY 10064555 Ki = 110 nM T47941 C69SBR 10068047 IC50 = 24000 nM T47941 C2L8MI 10068486 IC50 = 0.7943 nM T47941 CD3RL7 10070821 IC50 = 1 nM T47941 C7Q1DI 10071094 IC50 = 8 nM T47941 CJ4F8O 10072021 IC50 = 6 nM T47941 C5XQ9N 10072261 IC50 = 6 nM T47941 C4R1JU 10083346 Ki = 35800 nM T47941 C6PDN7 10083549 Ki > 200000 nM T47941 CBT1F3 10083557 Ki = 8200 nM T47941 C5P7AS 10083609 IC50 = 11000 nM T47941 CEG69D 10084247 Ki > 200000 nM T47941 CAX67L 10084334 IC50 = 3000 nM T47941 C2N4IZ 10084561 Ki = 0.54 nM T47941 C4X6DJ 10085014 Ki = 53000 nM T47941 C9R1JH 10085058 Ki = 136000 nM T47941 C8T3LV 10090103 IC50 = 1930 nM T47941 CP8I5O 10093297 IC50 = 24000 nM T47941 CUJX54 10094201 IC50 = 3.2 nM T47941 C7PU8W 10094320 IC50 = 30 nM T47941 CED4Z0 10094457 IC50 = 5.012 nM T47941 CS4QG0 10095269 IC50 = 3700 nM T47941 C61QRH 10096810 IC50 = 54000 nM T47941 C1OP0N 10105427 Ki = 27300 nM T47941 CFA3X7 10107643 Ki = 92400 nM T47941 CK5C9Z 10119563 IC50 = 15 nM T47941 C1EVS3 10119564 IC50 = 0.21 nM T47941 C3E4UM 10120032 IC50 = 1.7 nM T47941 CQ58PI 10130484 IC50 > 1000000 nM T47941 C8V1JR 10132419 IC50 = 1 nM T47941 CD5M9E 10133035 IC50 = 66 nM T47941 CH5EI6 10134821 IC50 = 6.2 nM T47941 C2YZ4H 10144464 IC50 = 0.7 nM T47941 CZG5Y6 10145190 IC50 = 1.4 nM T47941 C4F9HJ 10145470 IC50 = 0.6 nM T47941 C0XA4H 10151715 IC50 = 82 nM T47941 CVY3M2 10154549 IC50 > 100 nM T47941 C90GHX 10155377 IC50 = 0.18 nM T47941 COP10C 10156136 IC50 > 300 nM T47941 CO8NM5 10156864 IC50 > 1000 nM T47941 CBSM54 10157887 IC50 = 34 nM T47941 C7D5IT 10158829 IC50 = 52 nM T47941 C4NP8U 10167862 IC50 = 0.9 nM T47941 C8V2PN 10168172 IC50 = 1.4 nM T47941 CGA94F 10171570 IC50 = 500 nM T47941 C5WO3U 10171655 IC50 = 251.19 nM T47941 CACE30 10177300 IC50 = 2500 nM T47941 CS9W6X 10178224 IC50 > 1000 nM T47941 C3X9DK 10183196 IC50 = 31 nM T47941 CUXV40 10183769 IC50 = 1.6 nM T47941 CG81AB 10184563 IC50 = 1.995 nM T47941 CY9HS7 10185841 IC50 = 0.26 nM T47941 CYO0N7 10187078 IC50 = 1.5 nM T47941 CKX0P3 10189203 IC50 = 1.3 nM T47941 CI2A5S 10193005 IC50 = 1300 nM T47941 CS5TJ2 10193093 IC50 = 500 nM T47941 CVUZ36 10195164 IC50 = 7.8 nM T47941 CQ28MK 10198863 Ki = 14300 nM T47941 CE5LH4 10199681 IC50 = 19 nM T47941 C8DA4F 10200231 IC50 = 5.9 nM T47941 C18GTA 10201551 IC50 = 0.051 nM T47941 C61CZK 10205978 IC50 = 11 nM T47941 C6JHB3 10210431 IC50 = 0.8 nM T47941 CPU09I 10210579 IC50 = 0.93 nM T47941 CGMH76 10211390 IC50 = 0.2 nM T47941 CT6S9Y 10211456 IC50 = 0.4 nM T47941 CB35LH 10214932 IC50 = 790 nM T47941 C6B8VD 10221819 IC50 = 0.91 nM T47941 C1T3FV 10222690 IC50 > 30 nM T47941 C8DRL3 10232061 IC50 = 0.9 nM T47941 CX9LV3 10232106 IC50 = 0.2 nM T47941 CZ1Y8D 10232923 IC50 > 100000 nM T47941 C0TD1V 10236397 IC50 = 630 nM T47941 C6CN3D 10236419 IC50 = 320 nM T47941 C4R8YW 10236511 IC50 = 320 nM T47941 CSFU89 10243194 Ki = 32300 nM T47941 C2FE8T 10244649 Ki = 22300 nM T47941 C1XL2R 10247726 IC50 = 19000 nM T47941 CP8B1O 10248638 IC50 = 327 nM T47941 C7MQZ1 10249183 IC50 = 23 nM T47941 C0J3TC 10250722 IC50 = 300 nM T47941 C3AFN6 10250999 IC50 = 14000 nM T47941 CRK1U0 10252045 IC50 = 52000 nM T47941 CD8QY2 10253933 IC50 = 6.4 nM T47941 CI5Y3F 10254618 IC50 = 0.88 nM T47941 C7A9KM 10264889 Ki = 48700 nM T47941 CJQ89G 10266192 IC50 = 400 nM T47941 C7MR8P 10267945 IC50 = 4.7 nM T47941 C7RH4B 10270013 IC50 = 151 nM T47941 C5T9IR 10282859 IC50 = 0.2 nM T47941 CJ5KF2 10291951 IC50 = 0.29 nM T47941 CKR74B 10292282 IC50 = 7100 nM T47941 CECW14 10301548 IC50 = 0.12 nM T47941 CD83PR 10316172 IC50 = 348 nM T47941 CIPN48 10316358 IC50 = 37000 nM T47941 C3XV0B 10316470 IC50 = 81 nM T47941 CQ52HV 10316764 IC50 = 7000 nM T47941 CR72ZG 10317735 IC50 = 14 nM T47941 CH4AV8 10317875 IC50 = 48000 nM T47941 CI5Z3C 10317916 IC50 = 2400 nM T47941 CJV83M 10318617 IC50 = 2 nM T47941 C36AGZ 10321525 IC50 = 6500 nM T47941 C86USM 10326035 IC50 = 0.3162 nM T47941 CYM1D2 10330676 Ki = 28700 nM T47941 CAB62F 10332201 Ki = 16500 nM T47941 C07WRP 10333140 Ki = 72700 nM T47941 CRJW04 10334696 IC50 = 16000 nM T47941 CNEH87 10337932 IC50 = 40 nM T47941 C30JKP 10338622 Ki = 33 nM T47941 CLGA31 10341377 IC50 = 239 nM T47941 CP1M5H 10342086 IC50 = 4000 nM T47941 CMJG73 10342601 IC50 = 7100 nM T47941 CK05FV 10343476 IC50 = 37000 nM T47941 C6CBL3 10344500 IC50 = 23.3 nM T47941 C32IUF 10344870 IC50 = 24000 nM T47941 CJ7YZ9 10345293 IC50 = 1400 nM T47941 CA18KO 10347662 IC50 = 23000 nM T47941 C61OYX 10348848 IC50 = 42000 nM T47941 CC4W3M 10349233 IC50 = 5400 nM T47941 CR7TL0 10354640 Ki = 14600 nM T47941 C4ARN8 10355485 Ki = 119000 nM T47941 CQD9O7 10355498 IC50 = 37000 nM T47941 CCQ79O 10376254 Ki = 13200 nM T47941 C68BAQ 10376678 Ki = 23800 nM T47941 CK0J5U 10377117 Ki = 61400 nM T47941 C63XFI 10377425 Ki = 30800 nM T47941 CQ8Z9D 10378028 Ki = 29900 nM T47941 CW63NE 10378112 Ki = 13000 nM T47941 CYK1L7 10378132 Ki = 30100 nM T47941 CR35FX 10378878 IC50 = 19000 nM T47941 C5L7PZ 10378908 Ki > 200000 nM T47941 C2H9SE 10380126 IC50 = 8000 nM T47941 C0J7OV 10382041 IC50 = 10000 nM T47941 C8RYK7 10383026 IC50 = 2 nM T47941 CED0T9 10384709 IC50 = 341 nM T47941 C4FU9Q 10391767 IC50 = 700 nM T47941 C9-APR-07 10394586 IC50 = 20000 nM T47941 C4E1JH 10399896 Ki > 200000 nM T47941 C7LG8M 10400587 Ki > 200000 nM T47941 CI8B3P 10401473 IC50 = 6000 nM T47941 C6E0PG 10401818 IC50 = 9000 nM T47941 C0ADP3 10404378 IC50 = 41000 nM T47941 CRP4W3 10407214 IC50 = 800 nM T47941 CP8ZV5 10408375 IC50 = 3300 nM T47941 CU32AZ 10411395 IC50 = 0.631 nM T47941 CQUE27 10413015 IC50 = 45000 nM T47941 CP26NS 10422980 Ki = 9000 nM T47941 C0ZLB5 10423102 IC50 = 6000 nM T47941 C5HMX2 10428149 IC50 = 8100 nM T47941 CEOK50 10428730 IC50 = 12.59 nM T47941 CZ79QS 10430178 IC50 = 447 nM T47941 CEB7W1 10431107 IC50 = 2 nM T47941 C3WG2D 10432384 IC50 = 1 nM T47941 C82BMJ 10435245 IC50 = 0.35 nM T47941 CS0H3Z 10436258 IC50 = 0.51 nM T47941 C7HNX4 10445504 Ki = 20700 nM T47941 CZ8IC4 10448177 IC50 = 145 nM T47941 CU2HN6 10450290 IC50 = 51 nM T47941 CD09NL 10451631 IC50 = 541 nM T47941 CY95ME 10451799 IC50 = 824 nM T47941 C30WKM 10452355 IC50 = 719 nM T47941 CY4O0K 10452443 IC50 = 6900 nM T47941 C4LOK1 10454517 IC50 = 3300 nM T47941 CHQ38X 10455790 IC50 > 100000 nM T47941 CH2B6U 10455813 IC50 = 3800 nM T47941 CJM3L8 10456205 IC50 = 4.1 nM T47941 CR04LJ 10456913 IC50 = 44000 nM T47941 C9SHN7 10456942 IC50 = 5.2 nM T47941 CNW1O6 10467827 Ki = 46000 nM T47941 C2DEO3 10472374 IC50 = 65 nM T47941 CUD91J 10475033 IC50 = 34.99 nM T47941 CF0I6O 10479155 IC50 = 18000 nM T47941 C5CI3G 10479468 IC50 = 50 nM T47941 CA24TW 10491646 IC50 = 18000 nM T47941 C68VBD 10492653 IC50 = 49000 nM T47941 C3PKX6 10492654 IC50 = 4700 nM T47941 C5JPK7 10494678 EC50 = 2100 nM T47941 C4ZEI2 10495633 IC50 = 340 nM T47941 C7MFE0 10496166 IC50 = 420 nM T47941 C2OP8L 10497499 IC50 = 6300 nM T47941 C0P8OE 10500549 IC50 = 1940 nM T47941 C2W8OK 10501235 IC50 = 670 nM T47941 C14ITW 10502542 IC50 = 500 nM T47941 CMR6A4 10504383 IC50 = 200 nM T47941 C4CN0V 10508072 IC50 > 100000 nM T47941 CW7T6I 10515565 IC50 = 5100 nM T47941 CAWG05 10518739 IC50 = 1100 nM T47941 C86TDR 10522847 IC50 = 6040 nM T47941 CPWU60 10524067 IC50 = 40000 nM T47941 CPC16Z 10525153 IC50 = 130 nM T47941 CH4LZ1 10525677 IC50 = 690 nM T47941 CR8SN9 10526455 IC50 = 500 nM T47941 CZ6T2C 10536740 IC50 = 3100 nM T47941 CCG53Q 10541661 IC50 = 40000 nM T47941 CI7RY2 10542997 IC50 = 160 nM T47941 CLI1R7 10543311 IC50 = 6000 nM T47941 CAH2J6 10543697 IC50 = 1180 nM T47941 CQG9S1 10545255 IC50 = 25.2 nM T47941 C6M0ZQ 10545256 IC50 = 840 nM T47941 CDS4I1 10548443 IC50 = 360 nM T47941 C7T6YL 10548964 IC50 = 2800 nM T47941 C8TQ2B 10550635 Ki > 10000 nM T47941 CREU64 10551233 Ki = 45 nM T47941 C7ID5Q 10552011 IC50 = 1600 nM T47941 CMK39Q 10553487 IC50 = 200 nM T47941 CQW79N 10554042 IC50 = 5000 nM T47941 C4V8OI 10563356 IC50 = 39000 nM T47941 C5WMZ0 10563923 IC50 = 2300 nM T47941 CYUJ54 10564633 IC50 = 1000 nM T47941 C1R0HE 10567025 IC50 = 23000 nM T47941 CKUS20 10567758 IC50 = 750 nM T47941 C7K1QW 10571952 IC50 = 10500 nM T47941 CL7MR0 10572058 IC50 = 1800 nM T47941 CPF0R5 10572544 IC50 = 500 nM T47941 CYA19Q 10575041 IC50 = 4200 nM T47941 CWLQ30 10575043 IC50 = 3100 nM T47941 CY9P5W 10575733 IC50 = 5 nM T47941 C9ZFG7 10576010 IC50 = 1.3 nM T47941 C8V2KW 10576728 IC50 = 2700 nM T47941 CFY5J3 10576937 IC50 = 700 nM T47941 C20EPT 10577926 IC50 = 90 nM T47941 C7Z9YF 10579873 IC50 > 100000 nM T47941 CS5WL7 10589452 IC50 = 120 nM T47941 C3Y8JH 10590134 IC50 = 900 nM T47941 CZ3K8G 10591652 IC50 = 1200 nM T47941 CL4V5Z 10592156 IC50 = 150 nM T47941 C85MVT 10592818 IC50 = 3960 nM T47941 C1DI0R 10592954 Ki > 10000 nM T47941 CTCI60 10593194 IC50 = 34 nM T47941 CW0LN4 10593644 IC50 = 2300 nM T47941 CX2VD5 10594629 IC50 = 160 nM T47941 C5VX9F 10594814 IC50 = 567 nM T47941 C91UYR 10594887 IC50 = 84700 nM T47941 C4AH6Q 10596608 Ki = 3 nM T47941 CMNU92 10602385 IC50 = 80 nM T47941 CJ7CU4 10603606 IC50 = 0.9 nM T47941 CUTK97 10610142 IC50 = 14000 nM T47941 C8LT6P 10611956 IC50 = 7400 nM T47941 C5LVM2 10613420 IC50 = 13000 nM T47941 C1VZH9 10615487 IC50 = 1650 nM T47941 C0V1JY 10619481 IC50 = 20300 nM T47941 CPH0I1 10619533 IC50 = 300 nM T47941 CDO2C3 10619709 IC50 = 84900 nM T47941 C2WGV0 10620380 Ki = 10 nM T47941 CK3GR5 10624131 IC50 = 40 nM T47941 CFU29T 10625066 Ki = 1700 nM T47941 C31DUL 10625774 IC50 = 20 nM T47941 C1O4KV 10626842 IC50 > 100000 nM T47941 C25WRZ 10627119 IC50 = 0.55 nM T47941 C1JH0T 10639269 IC50 = 2500 nM T47941 CCB7D3 10639948 IC50 = 1500 nM T47941 CF1UR8 10640268 IC50 = 1500 nM T47941 CR7YM6 10641149 IC50 = 39 nM T47941 C4QRS6 10641529 Ki = 224 nM T47941 CB3R6M 10644497 IC50 = 16200 nM T47941 CZ5RG6 10646132 IC50 = 10800 nM T47941 CUZN30 10646721 IC50 = 700 nM T47941 CNK65G 10646809 IC50 = 70 nM T47941 CKNA14 10648008 IC50 = 0.68 nM T47941 CV2DE4 10648088 IC50 = 12 nM T47941 C0I4FA 10648358 IC50 = 330 nM T47941 CP8UX9 10649414 IC50 = 300 nM T47941 CE65JO 10650764 IC50 > 100000 nM T47941 CP2B0V 10660654 IC50 = 600 nM T47941 CY25HA 10661817 IC50 = 1100 nM T47941 C8KWM5 10663015 IC50 = 57000 nM T47941 CP1CJ3 10663161 IC50 = 29000 nM T47941 CP13SC 10663562 IC50 = 8100 nM T47941 C4R6LY 10664248 IC50 = 320 nM T47941 CD0NZ8 10664379 Ki = 100 nM T47941 CO03KC 10664439 IC50 = 221 nM T47941 CRA3W1 10667701 IC50 = 650 nM T47941 C09ROH 10668502 IC50 = 500 nM T47941 CC1S2F 10669014 Ki = 86 nM T47941 C4HJS1 10669027 IC50 = 9000 nM T47941 CB9Y7A 10669693 IC50 = 80 nM T47941 C9FR7P 10674875 IC50 > 100000 nM T47941 C2Y5HF 10675032 IC50 = 0.16 nM T47941 C6T4ZW 10687037 IC50 = 600 nM T47941 C5KXY7 10688351 EC50 = 2000 nM T47941 CNXT82 10689417 IC50 = 48 nM T47941 C47IFQ 10690189 IC50 = 1080 nM T47941 C28ZLH 10690190 IC50 = 490 nM T47941 CHB93E 10690761 IC50 > 200000 nM T47941 C84TDF 10691766 IC50 = 4700 nM T47941 CV6WT3 10692240 IC50 > 30000 nM T47941 C6LR4V 10694878 IC50 = 4700 nM T47941 C4U5VO 10695964 IC50 > 100000 nM T47941 CV0H5I 10696630 IC50 = 6200 nM T47941 C1B3WP 10696971 IC50 = 200 nM T47941 CI6ON5 10698519 IC50 = 0.49 nM T47941 C40GRD 10704663 IC50 = 11000 nM T47941 C23WGX 10706416 IC50 = 1900 nM T47941 C59SWD 10709216 IC50 = 5000 nM T47941 CG1AH4 10710468 IC50 = 63 nM T47941 C8CM0J 10711062 IC50 = 2700 nM T47941 C2GL3A 10714610 IC50 = 3000 nM T47941 C8UHE3 10717022 IC50 = 14000 nM T47941 CDMP96 10717370 IC50 = 50 nM T47941 CB82IG 10718103 Ki = 20 nM T47941 CEW0L8 10718244 IC50 = 2600 nM T47941 CU53RA 10718426 IC50 = 1400 nM T47941 CJ8EA6 10718949 IC50 = 1.2 nM T47941 CCI8R7 10729204 IC50 = 20000 nM T47941 CF7L2E 10732847 IC50 = 600 nM T47941 CC5X3R 10734134 IC50 = 660 nM T47941 CS2ZA3 10734331 IC50 = 1300 nM T47941 C5IKL9 10734997 IC50 = 1400 nM T47941 C8KVY9 10739717 IC50 = 750 nM T47941 CHVA02 10741072 IC50 = 2500 nM T47941 C2CG3U 10741142 Ki = 10 nM T47941 CGPA27 10742867 IC50 = 5900 nM T47941 CO39UQ 10744528 IC50 = 200 nM T47941 CJE9I8 10756115 IC50 = 1760 nM T47941 CIJ3H8 10757343 IC50 = 1640 nM T47941 CDPZ05 10758281 IC50 = 1100 nM T47941 CD5U4C 10759471 IC50 = 65000 nM T47941 CIQS47 10760137 IC50 = 178 nM T47941 CIW3A5 10760231 IC50 = 890 nM T47941 CLEG16 10761206 IC50 = 9000 nM T47941 CCE7H1 10761482 IC50 = 740 nM T47941 CINX82 10763354 IC50 = 20000 nM T47941 CB59DK 10764834 IC50 = 83 nM T47941 C3R8TI 10764856 IC50 = 760 nM T47941 CFJL61 10768238 IC50 = 0.2 nM T47941 C8QTA9 10768653 IC50 = 14 nM T47941 C51XRM 10776762 IC50 = 82000 nM T47941 C35YPM 10779997 IC50 = 16000 nM T47941 CO08EH 10780064 IC50 = 6700 nM T47941 CSN64H 10783300 IC50 = 2500 nM T47941 CEV60G 10783489 IC50 = 1000 nM T47941 CIN4A9 10783989 IC50 = 9000 nM T47941 C0GWH2 10783990 IC50 = 270 nM T47941 CI63NV 10784110 IC50 = 15700 nM T47941 CC4FE3 10784906 IC50 = 46 nM T47941 CKEV02 10786459 IC50 = 4000 nM T47941 C2THL7 10786618 IC50 = 1420 nM T47941 CQMF39 10787820 IC50 = 700 nM T47941 CLM42P 10788651 IC50 = 5000 nM T47941 CIJ76W 10789320 IC50 = 70 nM T47941 C92SMD 10789583 IC50 = 200 nM T47941 CHU2X8 10804455 IC50 = 3930 nM T47941 C59PSC 10805061 IC50 = 520 nM T47941 C9YFH4 10805458 IC50 = 3000 nM T47941 C79LJD 10807715 IC50 = 2240 nM T47941 CZV6R8 10808709 Ki = 37 nM T47941 C24LPM 10810360 IC50 = 26000 nM T47941 C9BGF7 10810371 IC50 = 460 nM T47941 CAF1X8 10812634 IC50 = 4200 nM T47941 CW07PN 10814053 IC50 = 200 nM T47941 CA9UW6 10816539 IC50 = 0.7 nM T47941 C4T8PS 10816641 IC50 > 100000 nM T47941 C49GKH 10826458 IC50 = 900 nM T47941 CG5M7O 10827879 IC50 = 1500 nM T47941 CKX2U7 10828701 IC50 = 160 nM T47941 CZ1I7Q 10828930 IC50 = 80 nM T47941 CT8AK4 10830480 IC50 = 1000 nM T47941 COHP57 10833764 IC50 = 20500 nM T47941 CO3EI8 10834255 IC50 = 140 nM T47941 C8HY0A 10835448 IC50 = 9000 nM T47941 CT2F6P 10835916 IC50 = 16000 nM T47941 C0QY8J 10837144 IC50 = 100 nM T47941 CIM93S 10840180 IC50 = 30 nM T47941 CR50XV 10841036 IC50 = 40 nM T47941 CQWL18 10852535 IC50 = 800 nM T47941 CCM2Y6 10853678 IC50 = 700 nM T47941 CE3H7M 10861002 IC50 = 2511.89 nM T47941 CPI5E6 10861494 IC50 = 79.43 nM T47941 CN4Y7B 10861789 IC50 = 25.12 nM T47941 C2O4TN 10862396 IC50 = 10 nM T47941 C5AYZ1 10871243 IC50 = 15.85 nM T47941 CSR0L6 10872703 IC50 = 2.512 nM T47941 CR4S0Q 10873246 IC50 = 19.95 nM T47941 CCV4L0 10873945 IC50 = 2.512 nM T47941 C3T4WD 10874925 IC50 = 7.943 nM T47941 CJ9H3C 10882487 IC50 = 12.59 nM T47941 C1N0WI 10882759 IC50 = 2511.89 nM T47941 CDF81X 10884865 IC50 = 0.631 nM T47941 C19DEY 10885064 IC50 = 6.31 nM T47941 CNG12D 10893436 IC50 = 1258.93 nM T47941 CV96UP 10894187 IC50 = 25.12 nM T47941 CR2I7H 10895319 IC50 > 10000 nM T47941 CU8A0Q 10895444 IC50 = 25.12 nM T47941 CE4O8T 10896876 IC50 = 10 nM T47941 CRJ5T9 10897006 IC50 = 0.3162 nM T47941 C0RTU9 10897531 IC50 = 3600 nM T47941 CW5EQ0 10903429 IC50 = 158.49 nM T47941 C8MZ6X 10904468 IC50 = 316.23 nM T47941 CO74IZ 10904782 IC50 = 316.23 nM T47941 CJM92R 10913208 IC50 = 7943.28 nM T47941 C38MIR 10916705 IC50 = 100 nM T47941 C42XNF 10917977 IC50 = 7.943 nM T47941 C1OY2D 10925930 IC50 = 79.43 nM T47941 CO9UW2 10927731 IC50 = 10 nM T47941 CR51HN 10935039 IC50 = 794.33 nM T47941 C6MDJ7 10937944 IC50 = 100 nM T47941 C2Z9IU 10938708 IC50 = 0.3981 nM T47941 CJ2G8Y 10939029 IC50 = 12.59 nM T47941 C5UY2I 10940665 IC50 = 6.31 nM T47941 CQ5F0N 10946130 IC50 = 125.89 nM T47941 CRA5Q4 10960172 IC50 = 25.12 nM T47941 CU05DG 10960538 IC50 = 6.31 nM T47941 CAB1K0 10970216 IC50 = 3.162 nM T47941 CKI1O9 10971811 IC50 = 1.585 nM T47941 CE1MC0 10980260 IC50 = 79.43 nM T47941 C9Q2OD 10980802 IC50 = 158.49 nM T47941 CEL8Z1 10980894 IC50 = 1995.26 nM T47941 C58LJN 10981074 IC50 > 10000 nM T47941 C4WN1U 10990720 IC50 = 39.81 nM T47941 C5XSJ3 10992513 IC50 = 15.85 nM T47941 CIJ18K 10993154 IC50 = 4900 nM T47941 C64POJ 10993740 IC50 = 10 nM T47941 C05TWX 11002318 IC50 = 79.43 nM T47941 C5Q2BD 11003326 IC50 = 1584.89 nM T47941 C1R4NH 11004936 IC50 = 63.1 nM T47941 C6DJH7 11013242 IC50 = 7.943 nM T47941 C0J4AS 11014562 IC50 = 79.43 nM T47941 CO6W2Q 11015053 IC50 = 3.162 nM T47941 C3AC7X 11015442 IC50 = 2511.89 nM T47941 CR7C1N 11017676 IC50 = 7000 nM T47941 C5AK1I 11023941 IC50 = 25.12 nM T47941 C2WJ3R 11026201 IC50 = 0.5012 nM T47941 C0ZW6I 11035565 IC50 = 251.19 nM T47941 CEK01S 11044358 IC50 = 100 nM T47941 CYN92B 11045774 IC50 = 2.512 nM T47941 CAN39X 11046445 IC50 = 50.12 nM T47941 CQK2X3 11048850 IC50 = 10 nM T47941 CCY7A3 11048935 IC50 = 39.81 nM T47941 CN5H2U 11056941 IC50 = 199.53 nM T47941 C4N1QY 11058335 IC50 = 7.943 nM T47941 CY0C8X 11058336 IC50 = 10 nM T47941 C4MA1V 11058378 IC50 = 0.5012 nM T47941 CV32FU 11058928 IC50 = 50.12 nM T47941 CQI5O1 11067303 IC50 = 125.89 nM T47941 CM02BE 11068268 IC50 = 3.981 nM T47941 CX75UB 11068454 IC50 = 794.33 nM T47941 CQ1J5C 11069107 IC50 = 1.259 nM T47941 CE28QV 11071990 IC50 = 0.631 nM T47941 CL0VC4 11072016 IC50 = 1.995 nM T47941 CA34RC 11075802 IC50 = 316.23 nM T47941 C8DQ2J 11077061 IC50 = 5011.87 nM T47941 CX68HJ 11078960 IC50 = 1584.89 nM T47941 C0T1DG 11079584 IC50 = 10 nM T47941 CI2TS9 11079673 IC50 = 19.95 nM T47941 CKM8F3 11089540 IC50 = 15.85 nM T47941 C03JQR 11089927 IC50 = 0.631 nM T47941 C8RZM1 11091364 IC50 = 19.95 nM T47941 CG74CI 11093245 IC50 = 6100 nM T47941 C52UJQ 11099452 IC50 = 39.81 nM T47941 CVOP12 11100066 IC50 = 31.62 nM T47941 CT8GE9 11100924 IC50 = 7.943 nM T47941 CPT9N5 11101908 IC50 = 12.59 nM T47941 C4VJR8 11109680 IC50 = 398.11 nM T47941 CG8F9N 11110230 IC50 = 63.1 nM T47941 CJIQ41 11110952 IC50 = 10 nM T47941 CG7FV9 11113983 IC50 = 5.012 nM T47941 C3IL4V 11120191 IC50 = 158.49 nM T47941 C2IQ1P 11121006 IC50 = 1.259 nM T47941 CLKO79 11121365 IC50 = 39.81 nM T47941 C5J7LY 11122692 IC50 = 12.59 nM T47941 CR1IZ3 11122701 IC50 = 1 nM T47941 C79DAI 11122877 IC50 = 25.12 nM T47941 CQ4D5W 11124276 IC50 = 3.981 nM T47941 C24VFA 11125005 IC50 = 1700 nM T47941 C9U6XR 11131381 IC50 = 158.49 nM T47941 C8P5RW 11132999 IC50 = 10 nM T47941 C9QKB3 11143180 IC50 = 1.259 nM T47941 CWHP16 11143259 IC50 = 63.1 nM T47941 C62VXY 11143924 IC50 = 15.85 nM T47941 CC3P5B 11152883 IC50 = 9 nM T47941 CFS4X6 11153159 IC50 = 0.9 nM T47941 C26PHV 11174905 IC50 = 62 nM T47941 CH6RQ0 11175536 IC50 = 20 nM T47941 C9GI2H 11175537 IC50 > 10000 nM T47941 CGW4M0 11188281 IC50 = 9.7 nM T47941 CP0M7U 11197828 IC50 = 160 nM T47941 CDO3S9 11199145 IC50 = 12 nM T47941 CSZ57O 11201305 IC50 = 0.85 nM T47941 CVG6J9 11244170 IC50 = 8000 nM T47941 C8SR7Q 11269374 IC50 = 80 nM T47941 CQ3ZX7 11289015 IC50 = 36 nM T47941 CG84VR 11301381 IC50 = 76 nM T47941 C63MWU 11303207 IC50 = 29 nM T47941 C5XRF3 11313467 IC50 = 26 nM T47941 C1A2SR 11325366 IC50 = 62 nM T47941 CTVZ70 11360233 IC50 = 100 nM T47941 C4C9GW 11372218 IC50 = 60000 nM T47941 CREQ98 11373312 IC50 = 4300 nM T47941 CU9IY2 11414494 IC50 = 4000 nM T47941 C1C7MW 11416279 IC50 = 20 nM T47941 CPH6E4 11426917 IC50 > 100 nM T47941 C96ENC 11500187 IC50 > 10000 nM T47941 CTE9G8 11522527 IC50 > 10000 nM T47941 C4ZYH9 11547485 IC50 = 1400 nM T47941 C37CQD 11551759 IC50 = 360 nM T47941 C7YVO3 11565462 IC50 > 10000 nM T47941 CW7UH3 11594581 IC50 = 680 nM T47941 CW1P4Y 11623586 IC50 = 380 nM T47941 CX2J4H 11640100 IC50 = 130 nM T47941 CPT8H6 11667299 IC50 > 1 nM T47941 C1A0KG 11726102 IC50 = 3700 nM T47941 C1JEQ5 11727597 IC50 = 1584.89 nM T47941 C4BH6M 11728213 IC50 = 7943.28 nM T47941 C6CE9Y 11728673 IC50 = 501.19 nM T47941 CLR4X2 11729202 IC50 = 15.85 nM T47941 C2BQ9K 11729404 IC50 = 15.85 nM T47941 CMS65Z 11729480 IC50 = 125.89 nM T47941 CZ26AP 11740167 IC50 = 120 nM T47941 C0AKJ4 11742456 IC50 = 6100 nM T47941 CA26IK 11742611 IC50 = 51 nM T47941 CX8J5U 11742876 IC50 = 100000 nM T47941 CROY49 11754228 IC50 = 110 nM T47941 C26CKE 11754697 IC50 = 3700 nM T47941 C5V1UG 11754942 IC50 = 32 nM T47941 CC92YE 11755033 IC50 = 550 nM T47941 CFE7S1 11762426 IC50 = 15.85 nM T47941 C1K3JX 11764545 IC50 = 56000 nM T47941 C7DWY1 11775680 IC50 = 53000 nM T47941 CNR1K6 11783406 IC50 = 5011.87 nM T47941 CQ8Y6L 11793138 IC50 = 20000 nM T47941 CGA1F8 11794425 IC50 = 200 nM T47941 C54KPM 11794796 Ki = 550 nM T47941 CYX91E 11795941 IC50 = 4400 nM T47941 C7E8QN 11796403 IC50 = 36000 nM T47941 CYZS05 11798266 IC50 = 1700 nM T47941 C2SXZ1 11798380 IC50 = 1000 nM T47941 CYN78M 11808269 IC50 = 6309.57 nM T47941 C2UH3J 11824398 IC50 = 0.5012 nM T47941 CT94GH 11826581 IC50 = 7.943 nM T47941 C29HOL 11828590 IC50 = 750 nM T47941 CK2J5S 11834125 IC50 > 10000 nM T47941 C7ZR6O 11857713 IC50 = 33000 nM T47941 CU5FJ6 11857715 IC50 = 14000 nM T47941 CO9I0H 12016984 IC50 = 37000 nM T47941 CZAV59 12016985 IC50 = 14000 nM T47941 CZ4QA8 12016986 IC50 = 3000 nM T47941 C08RSO 12016987 IC50 = 1200 nM T47941 C4YOB9 12016988 IC50 = 2100 nM T47941 C0VW2U 12016989 IC50 = 2100 nM T47941 C9ZWE6 12016990 IC50 = 6400 nM T47941 C8UL5M 12016991 IC50 = 7000 nM T47941 C28HJD 12016992 IC50 = 10000 nM T47941 CCL4W3 12016993 IC50 = 700 nM T47941 CAB5E1 12016994 IC50 = 800 nM T47941 CYF3K5 12016995 IC50 = 24000 nM T47941 C2M1JS 12017108 IC50 = 1300 nM T47941 CO6FU3 12041814 IC50 = 6.3 nM T47941 C6XAM3 12041815 IC50 = 874.98 nM T47941 CTN68G 12041817 IC50 = 164 nM T47941 C03HEV 12041818 IC50 = 85.1 nM T47941 C6DUZ1 12088731 IC50 = 15 nM T47941 C8NSP2 12088732 IC50 = 100 nM T47941 C3LH5B 12088733 IC50 = 25 nM T47941 CDF9Y2 12088734 IC50 = 18 nM T47941 CN8J2G 12088735 IC50 = 46 nM T47941 CIFK59 12088736 Ki = 54 nM T47941 C6THL1 12088737 Ki = 75 nM T47941 C30ZYX 12088738 Ki = 24 nM T47941 CG3H6W 12088761 IC50 = 8.59 nM T47941 CQUM27 12088765 IC50 = 16.98 nM T47941 CE4T6Z 12108678 IC50 = 69.98 nM T47941 C70FYQ 12268244 IC50 > 1000000 nM T47941 CB62GV 12922953 IC50 = 20000 nM T47941 CNST15 13136110 IC50 = 2000 nM T47941 C2WIF9 13248011 IC50 = 21000 nM T47941 C0CTE6 13388130 IC50 = 20000 nM T47941 CXZ71F 13388132 IC50 = 2500 nM T47941 CJ84NU 13408793 IC50 = 87000 nM T47941 C7XBF6 13408794 IC50 = 328000 nM T47941 CBFR79 13408796 IC50 = 16000 nM T47941 CY8K5T 13408798 IC50 = 350000 nM T47941 CD7X0S 13408812 IC50 = 339000 nM T47941 C05NRS 13408814 IC50 = 432000 nM T47941 CIP1O0 13408815 IC50 = 295000 nM T47941 CMSZ83 13408818 IC50 = 428000 nM T47941 CA2YP5 13408820 IC50 = 610000 nM T47941 CEDH78 13606768 IC50 = 33000 nM T47941 C8CKM9 13663754 IC50 = 339000 nM T47941 CE7ZW5 13785415 IC50 = 760 nM T47941 CF37AR 13815974 IC50 = 30000 nM T47941 CR5YK7 13815975 IC50 = 65000 nM T47941 C7SA3B 13815976 IC50 > 100000 nM T47941 CXG87I 13815977 IC50 = 20000 nM T47941 CT5WM6 13815978 IC50 = 25000 nM T47941 CX28FE 13815979 IC50 = 29000 nM T47941 CS31ZM 13815980 IC50 = 40000 nM T47941 CGA1Y9 13815981 IC50 = 7000 nM T47941 CC60WE 13815982 IC50 = 19000 nM T47941 CN4R7A 13815983 IC50 = 4000 nM T47941 C9X4EU 13815984 IC50 = 73000 nM T47941 CRPT87 13815985 IC50 = 2000 nM T47941 CV7FA6 13815986 IC50 = 2000 nM T47941 CFM6I4 13815987 IC50 = 49000 nM T47941 C1VWC9 13815990 IC50 = 27000 nM T47941 C6LN0I 13815991 IC50 = 15000 nM T47941 CWV0I6 13815992 IC50 = 30000 nM T47941 C9KR5X 13815995 IC50 > 100000 nM T47941 CF72VQ 14102450 IC50 = 400000 nM T47941 C3IYU7 14102465 IC50 = 3600 nM T47941 CB1LT4 14102469 IC50 = 10000 nM T47941 CO6I3H 14102471 IC50 = 30000 nM T47941 COWI58 14102485 IC50 = 29000 nM T47941 CY90SH 14180598 IC50 = 16 nM T47941 CT42IB 14180604 IC50 = 18500 nM T47941 CC9IM2 14180612 IC50 = 430 nM T47941 CJ5H6C 14180614 IC50 = 9.3 nM T47941 C7E5IH 14180616 IC50 = 63 nM T47941 CCX8J5 14180619 IC50 = 470 nM T47941 CPX1E4 14180621 IC50 = 8 nM T47941 C8TG5A 14180623 IC50 = 52 nM T47941 C14QKR 14180625 IC50 = 52 nM T47941 CI0M3V 14180628 IC50 = 100 nM T47941 CRSF89 14180630 IC50 = 120 nM T47941 CFBJ57 14180632 IC50 = 60 nM T47941 CO1H5A 14180633 IC50 = 3100 nM T47941 CMF30H 14208192 IC50 > 100000 nM T47941 CK29BD 14212369 IC50 = 150000 nM T47941 C9MT6X 14537151 IC50 = 96000 nM T47941 CYBE06 14537153 IC50 = 30000 nM T47941 CDX89G 14537155 IC50 = 22000 nM T47941 C2UKD7 14537156 IC50 = 400000 nM T47941 C1NLE9 14537157 IC50 = 34000 nM T47941 CU7R9N 14537158 IC50 = 16000 nM T47941 C92IFL 14537161 IC50 > 1000000 nM T47941 CC80NA 14537162 IC50 = 17000 nM T47941 CC8XP4 14537163 IC50 = 58000 nM T47941 CKPZ87 14537164 IC50 > 1000000 nM T47941 C94KCN 14537165 IC50 > 1000000 nM T47941 CB5S7X 14537166 IC50 = 13000 nM T47941 C8PLW7 14537167 IC50 = 18000 nM T47941 C7BDL8 14537168 IC50 = 24000 nM T47941 C30SCM 14537169 IC50 = 46000 nM T47941 CYWH06 14537170 IC50 > 1000000 nM T47941 CQM2P1 14537171 IC50 = 34000 nM T47941 CXZY62 14537172 IC50 = 25000 nM T47941 CW4J1E 14537173 IC50 = 19000 nM T47941 C42MOG 14537181 IC50 = 220000 nM T47941 C1RM0A 14537182 IC50 = 138000 nM T47941 C2ZX8H 14756622 IC50 = 500 nM T47941 CW3P1X 14803281 IC50 = 33000 nM T47941 C2X6HQ 14803339 IC50 = 33000 nM T47941 CIK71M 14836119 IC50 = 8900 nM T47941 CK3ZP8 14963574 IC50 = 170 nM T47941 CL2FY7 15192730 Ki = 159 nM T47941 C1YO3J 15294417 IC50 = 21000 nM T47941 CZ3P9I 15384033 IC50 = 410 nM T47941 C9AJP2 15435485 IC50 = 1700 nM T47941 CAC5H0 15606258 IC50 = 23000 nM T47941 CJW14P 15614030 Ki = 14100 nM T47941 C2W6VL 15614036 Ki = 12600 nM T47941 C6GXT7 15646969 Ki = 16400 nM T47941 C15FWY 15646970 Ki = 24100 nM T47941 CX08HC 15887290 IC50 = 120 nM T47941 CPQF96 15887291 IC50 = 26.98 nM T47941 CG3H7Y 15887293 IC50 = 53.95 nM T47941 C6QT8L 15931307 Ki = 26300 nM T47941 C5YDU4 15931309 Ki = 26000 nM T47941 C5BAJ3 15931313 Ki = 35000 nM T47941 C5BJ9K 16619271 IC50 = 100000 nM T47941 C9FN6T 17757112 IC50 = 20000000 nM T47941 C9LYS5 17757113 IC50 = 12000000 nM T47941 C3I6FH 17757114 IC50 > 20000000 nM T47941 C6EP0V 17757115 IC50 = 15000000 nM T47941 CET4G1 17757116 IC50 > 20000000 nM T47941 CXU2N8 17757118 IC50 = 13400000 nM T47941 CPS96I 17757119 IC50 = 12600000 nM T47941 CGB36A 17757120 IC50 = 14100000 nM T47941 C0LZ3H 17757121 IC50 > 20000000 nM T47941 C0YE8U 17757123 IC50 = 14100000 nM T47941 C2UQ0R 17757124 IC50 = 13400000 nM T47941 CK2R5T 17757125 IC50 = 19700000 nM T47941 CV79SK 17757126 IC50 > 20000000 nM T47941 CEO5W4 17757127 IC50 > 20000000 nM T47941 C5P8ZK 17757128 IC50 > 20000000 nM T47941 C2KMT0 17757129 IC50 > 20000000 nM T47941 CL3D6Y 17757130 IC50 = 11900000 nM T47941 CSBT76 17757131 IC50 > 20000000 nM T47941 C3ZH6X 17757132 IC50 = 112000 nM T47941 CM7UZ9 17757133 IC50 = 19700000 nM T47941 C6JW4M 17757134 IC50 = 13400000 nM T47941 C9YP8O 17757135 IC50 > 20000000 nM T47941 C27TQV 17757136 IC50 > 20000000 nM T47941 CLH36C 17757137 IC50 = 5300000 nM T47941 C09DZF 17757138 IC50 > 20000000 nM T47941 CC8K0Q 17757139 IC50 = 79000 nM T47941 CBZ15D 17757140 IC50 = 19600000 nM T47941 CUIO51 17757141 IC50 = 8000000 nM T47941 C58EBC 17757142 IC50 = 1700000 nM T47941 C8Z9SA 17757143 IC50 = 7500000 nM T47941 CEQ7X9 17757144 IC50 = 11900000 nM T47941 CF6V9I 17757145 IC50 > 20000000 nM T47941 CXFT59 17757146 IC50 = 10000 nM T47941 CVS6L9 17757147 IC50 = 8900000 nM T47941 CKW3E0 17757148 IC50 = 9000000 nM T47941 CS4HV9 17757149 IC50 = 6700000 nM T47941 C1RWA8 17757150 IC50 = 6900000 nM T47941 CIM84P 17757151 IC50 = 14100000 nM T47941 CJSI06 17757152 IC50 = 13400000 nM T47941 C3K4OA 17757153 IC50 = 13400000 nM T47941 C0TR1Q 17757154 IC50 = 9500000 nM T47941 C5E3NM 17757155 IC50 > 20000000 nM T47941 C0HPR1 17757156 IC50 = 12700000 nM T47941 C1K7EX 17757157 IC50 = 19600000 nM T47941 CR8UC7 17757158 IC50 = 50000 nM T47941 CAIR45 17757159 IC50 = 14100000 nM T47941 CY2B1S 17757160 IC50 = 14100000 nM T47941 C85SXY 17757161 IC50 > 20000000 nM T47941 C2XR7G 17757162 IC50 = 11200000 nM T47941 CZLQ38 17757163 IC50 = 4500000 nM T47941 C9DR5F 17757164 IC50 = 13400000 nM T47941 C37UGV 17757165 IC50 > 20000000 nM T47941 CC50HS 17757166 IC50 = 50000 nM T47941 CB8MR7 17757175 IC50 = 3200000 nM T47941 CI6S3B 17893099 IC50 = 1700 nM T47941 CBX29P 17989733 IC50 = 53 nM T47941 CT7J0R 18316653 IC50 = 120 nM T47941 CK8GI6 18332459 IC50 = 132 nM T47941 CXG1K2 18363133 IC50 = 55 nM T47941 C37BNA 18363136 IC50 = 49 nM T47941 C0KOW7 18363142 IC50 = 21 nM T47941 CP04KS 18363146 IC50 = 32 nM T47941 CLZD96 18363152 IC50 = 1500 nM T47941 CW3KB9 18363153 IC50 = 102 nM T47941 CK30ZO 18363159 IC50 = 89 nM T47941 CZU27R 18363164 IC50 = 50 nM T47941 CC0UV8 18363169 IC50 = 11 nM T47941 CR3CQ4 18363187 IC50 = 63 nM T47941 CH5IU9 18363209 IC50 = 31 nM T47941 CJGZ27 18363210 IC50 = 32 nM T47941 CWI2A9 18363212 IC50 = 260 nM T47941 C31LQZ 18363213 IC50 = 118 nM T47941 CE60WD 18363216 IC50 = 460 nM T47941 C3L6DU 18363223 IC50 = 140 nM T47941 CM4O9R 18381603 IC50 = 93.33 nM T47941 CTW2U6 18381613 IC50 = 30.2 nM T47941 C45TVJ 18381615 IC50 = 30 nM T47941 CI8WG0 18381641 IC50 = 112.2 nM T47941 CMCA10 18381646 Ki = 138 nM T47941 CKN72W 18381662 IC50 = 10 nM T47941 C7UT3G 18381674 IC50 = 51.29 nM T47941 CL5HK1 18381685 IC50 = 19 nM T47941 C8X9RW 18381692 IC50 = 38 nM T47941 C5VTK0 18393036 IC50 = 1 nM T47941 CF8QX2 18504823 IC50 = 186 nM T47941 C2LKM9 18504826 IC50 = 41.69 nM T47941 C1IOW8 18690934 IC50 = 0.7943 nM T47941 CZOT06 18690950 IC50 = 25.12 nM T47941 CYA3H7 18790040 IC50 = 580 nM T47941 CBN28Y 18790155 IC50 = 4600 nM T47941 CR78UH 18919373 IC50 = 1200 nM T47941 CL4GA8 18957476 IC50 = 500 nM T47941 CBW46P 19361840 IC50 = 68 nM T47941 C8A4YJ 19689634 IC50 = 1500 nM T47941 CVIC91 19690185 IC50 = 740 nM T47941 C21ZBP 20129307 IC50 = 10 nM T47941 C5L7AO 20346752 IC50 = 32000 nM T47941 CZ6GE2 20346768 Ki > 100000 nM T47941 C9DE6Y 20814950 IC50 = 450 nM T47941 C8PW2Q 21250943 IC50 = 2000 nM T47941 CX0Z1R 21360915 IC50 = 480 nM T47941 C3BL0G 21829352 IC50 = 4600 nM T47941 CN2YD9 21829362 IC50 = 50000 nM T47941 C7A1VL 21829707 IC50 = 29000 nM T47941 CF8ZP4 21840814 IC50 = 70 nM T47941 C48JRH 21840825 IC50 = 0.6 nM T47941 CMK42A 21952897 IC50 = 4.6 nM T47941 CG2P1F 21952923 IC50 > 1000 nM T47941 C5R0LQ 21952926 IC50 = 67 nM T47941 CMHF08 22083604 IC50 = 0.21 nM T47941 C34FLM 22083724 IC50 = 0.12 nM T47941 CWIT18 22083784 IC50 = 0.14 nM T47941 CM9RX0 22337173 IC50 = 398.11 nM T47941 CR4T9J 22337182 IC50 = 100 nM T47941 CE5T1U 22346826 IC50 = 6800 nM T47941 CJO7N9 22663188 IC50 = 2 nM T47941 C89JZG 22663193 IC50 = 5 nM T47941 CPEK75 22663199 IC50 = 27 nM T47941 C2G4OR 22663201 IC50 = 100 nM T47941 CRYQ07 22663228 IC50 = 25 nM T47941 CXLW87 22663231 IC50 = 45 nM T47941 CKY79J 22663238 IC50 = 4400 nM T47941 CO64GA 22663249 IC50 = 52 nM T47941 CI68PA 22663258 IC50 = 200 nM T47941 C56PAO 22663297 IC50 = 42 nM T47941 CR0QA1 22663307 IC50 = 23 nM T47941 CF8CA5 22663341 Ki = 187 nM T47941 CDG0R1 22663362 IC50 = 540 nM T47941 CY9XG3 22663364 IC50 = 2900 nM T47941 CM9EO4 22663370 IC50 = 450 nM T47941 CCH4D7 22734135 IC50 = 769.13 nM T47941 CM5H2P 23061661 IC50 = 1040 nM T47941 C97LAR 23061665 IC50 = 974 nM T47941 CD48PX 23218492 IC50 = 224 nM T47941 C0T4GY 23515911 IC50 = 6770 nM T47941 CD0F5Y 23672439 IC50 = 31.62 nM T47941 CZ8BQ6 24737709 IC50 = 22400 nM T47941 C4GUC1 24738493 IC50 = 261 nM T47941 CLH3G9 24738495 IC50 = 23 nM T47941 CCO8T6 24738496 IC50 = 77 nM T47941 C4H6WK 24810298 IC50 = 84000 nM T47941 C20VHK 24871823 IC50 = 3700 nM T47941 CAL48H 24883367 IC50 = 2 nM T47941 CPY8C0 24901352 IC50 = 0.53 nM T47941 CA37DH 25010445 IC50 = 570 nM T47941 CK7J6A 25010446 IC50 = 4400 nM T47941 CVN86W 25010447 IC50 = 6000 nM T47941 C7CWK1 25010450 IC50 = 6400 nM T47941 CAN21O 25010622 IC50 > 30000 nM T47941 C4YT9V 25147797 IC50 = 22 nM T47941 C0JHE6 25178111 IC50 = 100000 nM T47941 CR16QH 25178733 IC50 = 93000 nM T47941 C6BWC9 25178734 IC50 = 29000 nM T47941 CS17JC 25178735 IC50 = 60000 nM T47941 CY8J7K 25178736 IC50 = 71000 nM T47941 CF1RU9 25178737 IC50 = 24000 nM T47941 CQL8C0 25178738 IC50 = 100000 nM T47941 CS3W8X 25178918 IC50 = 720 nM T47941 C8ZD0X 25178920 IC50 = 430 nM T47941 C3B9ID 25178922 IC50 = 1900 nM T47941 C1GZ8X 25178923 IC50 = 2600 nM T47941 C3SG2C 25179111 IC50 = 1100 nM T47941 CA29CE 25179112 IC50 = 180 nM T47941 CRV0E8 25179115 IC50 = 40000 nM T47941 CMJ40D 25179281 IC50 = 5200 nM T47941 CTK06Q 25179476 IC50 = 2300 nM T47941 CNZM75 25179676 IC50 = 667 nM T47941 CQ6M3L 25179677 IC50 = 626 nM T47941 CWC1O2 25179678 IC50 = 350 nM T47941 C89JPH 25179679 IC50 = 44000 nM T47941 CGC01Z 25179875 IC50 = 82 nM T47941 CXF18O 25181027 IC50 = 100000 nM T47941 C8QMT0 25258345 IC50 = 820 nM T47941 C6D3YJ 30133545 IC50 = 600 nM T47941 CY8Q3T 44143467 IC50 > 20000000 nM T47941 C5QKJ1 44143468 IC50 > 20000000 nM T47941 C5X9AD 44209387 IC50 > 100000 nM T47941 C0ZKN1 44209388 IC50 > 100000 nM T47941 C5OB0R 44223559 IC50 = 1500 nM T47941 CSI24U 44223606 IC50 = 3700 nM T47941 C7Y0HI 44274612 IC50 = 110 nM T47941 CA6J8T 44274920 IC50 = 300 nM T47941 CVJE04 44276974 IC50 = 23000 nM T47941 C2MH7V 44279469 IC50 = 1100 nM T47941 CU0CH7 44279583 IC50 = 1300 nM T47941 CX89AE 44279648 EC50 = 200 nM T47941 CU8GE2 44279665 IC50 = 1500 nM T47941 C1OC5N 44280175 IC50 = 11000 nM T47941 C02PWF 44281897 IC50 = 500000 nM T47941 C9LV1F 44281955 IC50 = 800000 nM T47941 C9PHZ0 44288339 IC50 = 87.9 nM T47941 CQJX15 44288425 IC50 = 179.89 nM T47941 CJYF67 44288428 IC50 = 209.89 nM T47941 CM0Q3P 44288456 IC50 = 700 nM T47941 CW8I1T 44288506 IC50 = 10000 nM T47941 CSD8A2 44288553 IC50 = 439.54 nM T47941 C8XK0U 44288560 IC50 = 42.95 nM T47941 C3JDA0 44288639 IC50 = 289.73 nM T47941 CBT10V 44288640 IC50 = 480 nM T47941 CN4L0A 44288664 IC50 = 110 nM T47941 CJ1HT6 44288855 IC50 = 9.5 nM T47941 CV13MZ 44288878 IC50 = 1119.44 nM T47941 CT38HI 44289140 IC50 = 64 nM T47941 CAH30U 44289181 IC50 = 16 nM T47941 CH1TS5 44289182 IC50 = 5250 nM T47941 CMZ2O6 44289200 IC50 > 10000 nM T47941 C7WUJ2 44289459 IC50 = 564 nM T47941 CJ73FW 44289479 IC50 = 36 nM T47941 CWMI67 44289482 IC50 = 3030 nM T47941 C1L4ZU 44289489 IC50 = 295 nM T47941 C19EJM 44289515 IC50 = 14 nM T47941 CA52ED 44289521 IC50 = 280 nM T47941 C7GY8M 44289643 IC50 = 3600 nM T47941 CV9B2F 44289867 IC50 = 520 nM T47941 CANC98 44292198 IC50 = 0.5 nM T47941 CB5AY3 44293676 IC50 = 18000 nM T47941 C04AMH 44293703 IC50 = 1000 nM T47941 C93TWC 44294027 IC50 > 100000 nM T47941 CGS93T 44294544 IC50 = 1700 nM T47941 C64BWE 44294729 IC50 = 1200 nM T47941 CYU6L2 44294730 IC50 = 1000 nM T47941 CQ6F3Y 44294731 IC50 = 700 nM T47941 CIC45P 44294818 IC50 = 54000 nM T47941 CX32VT 44294906 IC50 = 1000 nM T47941 CB0CO4 44294974 Ki > 3700 nM T47941 CG47KS 44294992 Ki = 200 nM T47941 CX54OL 44295012 IC50 = 2000 nM T47941 CWTK85 44295026 IC50 = 500 nM T47941 CIS42L 44295159 IC50 = 2400 nM T47941 CEH82G 44295178 IC50 = 200 nM T47941 CNK73O 44295200 IC50 = 4600 nM T47941 CSEC93 44298012 Ki = 63900 nM T47941 CGR3B7 44298016 Ki = 260 nM T47941 CPU0S2 44298017 Ki = 1170 nM T47941 C9LQE5 44298054 Ki = 3690 nM T47941 CB5H8R 44298227 Ki = 220 nM T47941 C6MU7H 44298228 Ki = 172 nM T47941 CP5A9M 44298255 IC50 = 12 nM T47941 C6S4KU 44298440 Ki > 3745 nM T47941 CE5A3N 44298444 IC50 = 60 nM T47941 CS9B4H 44298484 IC50 = 25 nM T47941 C3TOH5 44298485 IC50 = 70 nM T47941 CZCF20 44301566 IC50 = 3400 nM T47941 C72WTZ 44301567 IC50 = 7100 nM T47941 C7OE6X 44301799 IC50 = 3600 nM T47941 CT6QN1 44301814 IC50 = 1200 nM T47941 CI80MC 44301836 IC50 = 1700 nM T47941 CV13JY 44301955 IC50 = 81 nM T47941 CC8PN0 44301959 IC50 = 103 nM T47941 CR76QT 44301964 IC50 = 71 nM T47941 C4LFB6 44308040 IC50 = 2.41 nM T47941 CXQT32 44308118 IC50 = 451.86 nM T47941 CRIZ14 44308285 IC50 = 319.89 nM T47941 CR1TN2 44308308 IC50 = 330.37 nM T47941 CZ9BG0 44308597 IC50 = 3400 nM T47941 CP5AZ7 44308638 IC50 = 150 nM T47941 CP6F1C 44311694 IC50 = 153 nM T47941 CW75QH 44312546 IC50 = 2.9 nM T47941 CL80RT 44314758 IC50 = 450 nM T47941 C3ID9H 44314916 IC50 = 100000 nM T47941 CC6F4N 44315110 IC50 = 50000 nM T47941 C0KT9E 44318468 IC50 = 630.96 nM T47941 C4RWG3 44318473 IC50 = 50.12 nM T47941 C05BHP 44318551 IC50 = 3.981 nM T47941 CJ5O6S 44318686 IC50 = 12.59 nM T47941 CW0XS1 44318693 IC50 = 25.12 nM T47941 C3L6AF 44319378 IC50 = 25.12 nM T47941 C76POF 44321935 IC50 = 900 nM T47941 CN8I5G 44321936 IC50 = 1800 nM T47941 CR1H2G 44322008 IC50 = 460 nM T47941 CHWX64 44322250 IC50 = 23000 nM T47941 C0B5UA 44322260 IC50 = 49000 nM T47941 C2G7YF 44322548 IC50 = 7800 nM T47941 CVK2G9 44322618 IC50 = 600 nM T47941 CBWY78 44322628 IC50 = 3000 nM T47941 CZ4UF7 44322638 IC50 = 1900 nM T47941 C4UJL8 44322650 IC50 = 10000 nM T47941 CAJO73 44322688 IC50 = 1500 nM T47941 CANB83 44322689 IC50 = 2000 nM T47941 C81DTK 44322707 IC50 = 24000 nM T47941 C19WBO 44322747 IC50 = 5000 nM T47941 C92KBQ 44322800 IC50 = 5200 nM T47941 C8S7CK 44322828 IC50 = 2500 nM T47941 CWE42S 44322842 IC50 = 3000 nM T47941 CK5RO3 44322844 IC50 = 500 nM T47941 C0WMF3 44322856 IC50 = 4000 nM T47941 CU5O8Z 44322857 IC50 = 6000 nM T47941 C8G0JI 44322864 IC50 = 5300 nM T47941 CKD9J3 44322865 IC50 = 9000 nM T47941 CR41FC 44323256 IC50 = 700 nM T47941 C05VLD 44323257 IC50 = 18000 nM T47941 C2-JAN-01 44323270 IC50 = 160000 nM T47941 CBP5I9 44323409 IC50 = 11000 nM T47941 C0XZ6H 44323410 IC50 = 400 nM T47941 CK5ZG3 44323424 IC50 = 2700 nM T47941 CFUB24 44323425 IC50 = 2300 nM T47941 CP5N9V 44323427 IC50 = 12000 nM T47941 C5IJQ8 44323428 IC50 = 500 nM T47941 CMFX02 44323504 IC50 = 800 nM T47941 C21UJZ 44323510 IC50 = 90000 nM T47941 C2FZS7 44323529 IC50 = 340 nM T47941 CCET86 44323543 IC50 = 2200 nM T47941 CAH1Q0 44323556 IC50 = 1400 nM T47941 CZ16IY 44324251 IC50 = 600 nM T47941 CCX9Z3 44324252 IC50 = 450 nM T47941 CQHB05 44324264 IC50 = 2540 nM T47941 CG6UT1 44324296 IC50 = 600 nM T47941 CYA3R9 44324299 IC50 = 36200 nM T47941 C2SLH8 44324331 IC50 = 603 nM T47941 C8M4WJ 44324373 IC50 = 500 nM T47941 CY5HZ7 44324390 IC50 = 30 nM T47941 C5KYV6 44324391 IC50 = 70 nM T47941 C5C4QX 44324507 IC50 = 57 nM T47941 C34YOB 44325316 IC50 = 45 nM T47941 CTKA30 44325479 IC50 = 28 nM T47941 C0J6RT 44330813 IC50 = 20000 nM T47941 CCLK42 44330913 IC50 = 110000 nM T47941 CG9O1R 44330960 IC50 > 20000 nM T47941 CUZK78 44330961 IC50 = 20000 nM T47941 CT2EB9 44330971 IC50 = 100000 nM T47941 CKC74R 44331037 IC50 = 2400 nM T47941 CD9N4L 44334251 IC50 = 24 nM T47941 C9RMD5 44334262 IC50 = 22 nM T47941 C2XE1N 44334271 IC50 = 7 nM T47941 CIPY56 44334272 IC50 = 14 nM T47941 C3W5OQ 44334291 IC50 = 46 nM T47941 CWTJ48 44334301 IC50 = 260 nM T47941 C25VFB 44334302 IC50 = 38 nM T47941 C92MFR 44334310 IC50 = 12 nM T47941 CGQJ50 44334340 Ki = 64 nM T47941 CSPH87 44334341 IC50 = 1400 nM T47941 CN7GX9 44334346 Ki = 393 nM T47941 CP6H3S 44334347 Ki = 225 nM T47941 CE09LF 44334393 IC50 = 16 nM T47941 CK7ZJ1 44334414 IC50 = 19 nM T47941 C7P8YK 44334422 IC50 = 20 nM T47941 CTG69B 44338110 IC50 = 250 nM T47941 CF0J4Q 44338111 IC50 > 300 nM T47941 CY3VQ8 44338541 IC50 = 97 nM T47941 CUX02O 44338550 IC50 > 300 nM T47941 CQ28VW 44338555 IC50 > 300 nM T47941 CSZ6M5 44338556 IC50 = 85 nM T47941 CX5D8G 44338611 IC50 > 100 nM T47941 CQ21KB 44338777 IC50 > 100 nM T47941 CJ65GD 44338778 IC50 > 100 nM T47941 CCOZ32 44339609 IC50 = 2200 nM T47941 CH9P3C 44348937 IC50 = 1800 nM T47941 CVA3O4 44348938 IC50 = 1250 nM T47941 CVW1P2 44348994 IC50 = 630 nM T47941 C5T6BV 44348995 IC50 = 960 nM T47941 C2Q9XZ 44349115 IC50 = 760 nM T47941 C5DKS3 44349135 IC50 = 1150 nM T47941 CS4QH0 44349295 IC50 = 650 nM T47941 C4GDB0 44352576 IC50 = 4700 nM T47941 C0WH4X 44352624 EC50 = 21000 nM T47941 CC3P1L 44352733 IC50 = 10000 nM T47941 C5QWL2 44352901 IC50 = 44 nM T47941 CP2ZH5 44352903 Ki = 4.3 nM T47941 CX7ST1 44352916 IC50 = 293 nM T47941 C10VJU 44352934 Ki = 210 nM T47941 CZJ4G1 44352945 Ki > 3745 nM T47941 CI60FZ 44352954 Ki = 337 nM T47941 CKEY07 44352955 IC50 = 6.3 nM T47941 CGYF87 44352984 IC50 = 1600 nM T47941 CG14PY 44352997 IC50 = 293 nM T47941 CN42LW 44353084 IC50 = 59 nM T47941 C73LEA 44353093 Ki = 787 nM T47941 C0Q4JO 44353102 IC50 = 123 nM T47941 CQZ21J 44353103 Ki = 367 nM T47941 C0MNA7 44353113 Ki = 43 nM T47941 C28ZFB 44353114 Ki = 80 nM T47941 C1EVC2 44353116 Ki = 274 nM T47941 CC4EI7 44353121 IC50 = 82 nM T47941 C2I0OQ 44353124 IC50 = 61 nM T47941 C7G0RE 44353125 IC50 = 401 nM T47941 CAP89V 44353133 Ki = 51 nM T47941 CX6W2U 44353156 IC50 = 137 nM T47941 CI7DW1 44353157 Ki = 470 nM T47941 C1FEJ6 44355478 Ki = 20 nM T47941 C7RX4E 44355596 Ki = 20 nM T47941 C7LN0W 44363056 IC50 = 9500 nM T47941 C71YUD 44363183 IC50 = 44000 nM T47941 CZX3H7 44364909 IC50 = 14000 nM T47941 C8HWG0 44364924 IC50 = 7900 nM T47941 C9YDX5 44364932 IC50 = 7600 nM T47941 CTZ40A 44365004 IC50 = 32000 nM T47941 C2WGA3 44365034 IC50 = 8600 nM T47941 CAM5B4 44365046 IC50 = 15000 nM T47941 CMX5H0 44365049 IC50 = 30000 nM T47941 CU2T5E 44365050 IC50 = 90000 nM T47941 C9FME0 44365068 IC50 = 74000 nM T47941 CA26VF 44365094 IC50 = 3300 nM T47941 CZ5V7K 44365144 IC50 = 3.7 nM T47941 C3M4YD 44365208 IC50 = 42000 nM T47941 CE0MT4 44365229 IC50 = 3800 nM T47941 C8XC2Q 44365265 IC50 = 107000 nM T47941 CEZS84 44365300 IC50 = 48 nM T47941 C4EYC2 44365329 IC50 = 66 nM T47941 CEZM67 44365330 IC50 = 140 nM T47941 CKE53Q 44365343 IC50 = 230 nM T47941 CV6H1T 44365386 IC50 = 47 nM T47941 C9HO0T 44365387 IC50 = 47 nM T47941 CEL9B6 44365476 IC50 = 62 nM T47941 C09ZIV 44365522 IC50 = 120 nM T47941 CZ28YH 44365523 IC50 = 120 nM T47941 CFVC04 44365547 IC50 = 23 nM T47941 CA3Z4H 44377154 IC50 = 3610 nM T47941 CQ71SK 44377233 IC50 = 1070 nM T47941 CWFJ24 44377249 IC50 = 5910 nM T47941 C3EP6H 44380311 IC50 = 52 nM T47941 CLMW27 44405467 IC50 = 1.2 nM T47941 CR05OY 44405507 IC50 = 8.3 nM T47941 C7OA9V 44405510 IC50 = 0.61 nM T47941 C6RFB5 44409461 IC50 = 630 nM T47941 C8H5WF 44409462 IC50 = 2000 nM T47941 CX7R9U 44409463 IC50 = 400 nM T47941 C1JN2W 44409556 IC50 = 4000 nM T47941 C48TAF 44409557 IC50 = 3200 nM T47941 CL1UM2 44409558 IC50 = 500 nM T47941 CI8UH3 44409576 IC50 = 790 nM T47941 C65LDN 44409651 IC50 = 630 nM T47941 C41BTQ 44409653 IC50 = 790 nM T47941 C7UE8I 44409654 IC50 = 790 nM T47941 CR5N4B 44409660 IC50 = 2000 nM T47941 CTH4U7 44409744 IC50 = 400 nM T47941 C1SNK8 44409745 IC50 = 400 nM T47941 C1DR6L 44409746 IC50 = 630 nM T47941 CU5PZ9 44409749 IC50 = 630 nM T47941 CLWK34 44409751 IC50 = 2000 nM T47941 CVUL24 44409754 IC50 = 400 nM T47941 CXQ1E6 44409755 IC50 = 1600 nM T47941 CSK9M0 44409759 IC50 = 1600 nM T47941 COZ39R 44409760 IC50 = 2500 nM T47941 C58LXG 44409765 IC50 = 3200 nM T47941 C5Y9MU 44409769 IC50 = 2500 nM T47941 CQI9A1 44409772 IC50 = 1600 nM T47941 CNJC24 44409787 IC50 = 1260 nM T47941 CN06AV 44409796 IC50 = 2000 nM T47941 CU4KQ2 44409797 IC50 = 4000 nM T47941 CWPZ82 44409937 IC50 = 790 nM T47941 CS6UR7 44409944 IC50 = 6300 nM T47941 C5VFP3 44409945 IC50 = 7900 nM T47941 CBXV64 44409956 IC50 = 2500 nM T47941 CUV53S 44409961 IC50 = 2000 nM T47941 C4XBR6 44409962 IC50 = 500 nM T47941 C4VZ5R 44409963 IC50 = 1000 nM T47941 CU64VF 44409965 IC50 = 2500 nM T47941 CAR61H 44409976 IC50 = 2000 nM T47941 CLT2Y3 44409977 IC50 = 6300 nM T47941 C48QIT 44409978 IC50 = 2500 nM T47941 CK46WN 44409981 IC50 = 2000 nM T47941 CY0F6E 44409982 IC50 = 1260 nM T47941 CV3U9L 44409995 IC50 = 250 nM T47941 CJT90I 44430454 IC50 = 3200 nM T47941 C8KO4X 44430461 IC50 = 5000 nM T47941 CEL85Z 44430462 IC50 = 630 nM T47941 C1WA3Q 44430464 IC50 = 2000 nM T47941 C7L8CO 44430466 IC50 = 1000 nM T47941 CJ6Z8U 44430467 IC50 = 50.12 nM T47941 CL0VG4 44430469 IC50 = 500 nM T47941 C9SQ4Y 44430470 IC50 = 4000 nM T47941 CFRQ71 44430472 IC50 = 790 nM T47941 CYQ0N1 44430473 IC50 = 2000 nM T47941 CQIA96 44430474 IC50 = 200 nM T47941 CSZ3H9 44457773 IC50 = 130 nM T47941 CC31TH 44461328 IC50 = 153 nM T47941 C57FAU 44461405 IC50 = 131 nM T47941 C57MZU 44461420 IC50 = 36 nM T47941 CR0KP5 44461430 IC50 = 85 nM T47941 C50ZNL 44461693 IC50 = 30 nM T47941 C1S4ZT 44461851 IC50 = 3.981 nM T47941 C5L6KP 44541346 IC50 = 3620 nM T47941 CPY3W6 44541483 IC50 = 3980 nM T47941 C4C9RI 44541606 IC50 = 1460 nM T47941 CIYL43 44541609 IC50 = 6700 nM T47941 C8F3UO 44562338 IC50 = 15.85 nM T47941 CA0G5Y 44565465 IC50 = 710 nM T47941 CAN70F 44577780 IC50 > 1 nM T47941 C3SL5Y 44591584 IC50 = 3400 nM T47941 C4ZXG2 44591585 IC50 > 10000 nM T47941 C7ZHR1 44591599 IC50 = 7700 nM T47941 CJ8RT3 44591600 IC50 = 1300 nM T47941 C2P7MK 44591614 IC50 = 2000 nM T47941 CB5M1J 44591615 IC50 = 2700 nM T47941 CG5H3Y 44591616 IC50 = 450 nM T47941 CJP30T 44591617 IC50 > 30000 nM T47941 C4HL9P 44755057 IC50 = 29000 nM T47941 C45ZVC 45258276 IC50 = 63 nM T47941 C2N9HA 45259270 IC50 = 150 nM T47941 C10TQI 45259276 IC50 = 31 nM T47941 CBKJ47 45259284 IC50 = 700 nM T47941 CSX9O6 45259293 IC50 = 30 nM T47941 C31FMT 45260180 IC50 = 121000 nM T47941 CCQ35I 45260248 IC50 = 53000 nM T47941 C3V5FJ 45260731 IC50 = 0.3 nM T47941 CH19WE 45260740 IC50 = 3 nM T47941 CM45BI 45260745 IC50 = 0.3 nM T47941 CM24BL 45260747 IC50 = 0.4 nM T47941 CN3A9L 45260753 IC50 = 2 nM T47941 CIT9E7 45260778 IC50 = 0.5 nM T47941 CSJZ49 45263853 IC50 = 190 nM T47941 CVSY51 45263858 IC50 = 17 nM T47941 C1Y9CW 45263914 IC50 = 15 nM T47941 CTEP18 45484024 IC50 = 10500 nM T47941 CX90YO 45484534 IC50 = 0.3 nM T47941 C0D2MN 46186792 IC50 > 10000 nM T47941 C0WRO9 46198713 IC50 > 10000 nM T47941 CXG34R 46199487 IC50 > 10000 nM T47941 CAL85J 46199794 IC50 = 6960 nM T47941 CI9EA4 46199799 IC50 = 3680 nM T47941 C26RJV 46200090 IC50 = 176 nM T47941 C5WND9 46200233 IC50 > 10000 nM T47941 CKIC45 46200238 IC50 > 10000 nM T47941 CS46AE 46200399 IC50 > 10000 nM T47941 C1S3BK 46200706 IC50 = 2920 nM T47941 C4P5QJ 46200709 IC50 = 70.8 nM T47941 CV8Y6W 46200711 IC50 > 10000 nM T47941 CK1N4X 46200728 IC50 > 1000 nM T47941 CH9FU8 46200877 IC50 > 1000 nM T47941 CEZ3V4 46200878 IC50 = 3670 nM T47941 CI1F5C 46239840 Ki >= 770 nM T47941 C26XVS 46240044 Ki >= 4793 nM T47941 CE4JU7 46842025 IC50 > 10000 nM T47941 CR8JC2 46842169 IC50 > 10000 nM T47941 CKAV30 46844770 IC50 = 75 nM T47941 C4DSX7 46844771 IC50 = 32 nM T47941 C3D9QG 46844772 IC50 = 59 nM T47941 C9MLV0 46878258 IC50 = 210 nM T47941 CM7VP4 46887175 IC50 = 385 nM T47941 C5YVK9 46887209 IC50 = 300 nM T47941 CD0L4E 46887237 IC50 = 237 nM T47941 CSL5W0 46887238 IC50 = 72 nM T47941 C61CMA 46887239 IC50 = 374 nM T47941 CD6F2Q 46887277 IC50 = 876 nM T47941 CK9YW6 46887278 IC50 = 757 nM T47941 C51GLW 46887280 IC50 = 1140 nM T47941 CDRL93 46887281 IC50 = 1200 nM T47941 CC4GV5 46887375 IC50 = 46 nM T47941 CWXA27 46887424 IC50 = 32 nM T47941 C7T2GX 46909057 IC50 = 9750 nM T47941 CZM3O9 49796282 IC50 = 35 nM T47941 CZS03D 50902030 Ki > 4274 nM T47941 CH2Z1E 50902289 Ki > 7100 nM T47941 C4HJL2 50902291 Ki > 7950 nM T47941 C6A1IU 50902549 Ki > 2000 nM T47941 C3Y2AV 50903255 Ki > 2000 nM T47941 CSHK08 52942937 IC50 = 0.2 nM T47941 CHY9P7 52945359 IC50 = 0.4 nM T47941 CST08G 52947776 IC50 = 0.4 nM T47941 CVF79G 52947777 IC50 = 0.2 nM T47941 CAT5L0 53323012 IC50 = 6000 nM T47941 CAL3I1 53326944 IC50 = 6000 nM T47941 C8CG9H 53703819 IC50 = 83 nM T47941 CTP54Y 54238057 IC50 = 350 nM T47941 C1AND4 56659469 IC50 = 6400 nM T47941 CGWH19 56662928 IC50 > 40000 nM T47941 CQT17K 56662929 IC50 = 510 nM T47941 CLMG01 56662930 IC50 = 220 nM T47941 CL1U3W 56666405 IC50 = 230 nM T47941 C5H9XA 56669821 IC50 > 5000 nM T47941 CIX9M0 56673307 IC50 = 150 nM T47941 CTY48D 56673902 IC50 = 1300 nM T47941 CEO42M 56676640 IC50 = 280 nM T47941 C2CRW3 56679969 IC50 = 0.57 nM T47941 CT8A6K 56683302 IC50 = 200 nM T47941 CGEV72 56834882 IC50 = 469 nM T47941 CC6ZD0 57390813 IC50 = 3770 nM T47941 CCP74G 57392635 IC50 = 982 nM T47941 C7EOQ2 57396104 IC50 = 8420 nM T47941 CB1C3G 57396105 IC50 = 4840 nM T47941 CAN16F 57397919 IC50 = 11900 nM T47941 CZ1F9G 57397920 IC50 = 342 nM T47941 C42TCU 57399123 IC50 = 2200 nM T47941 C7DJ9Q 57399527 IC50 = 1060 nM T47941 CVKR29 57399561 IC50 = 4340 nM T47941 C25ULW 57399562 IC50 = 1300 nM T47941 CP0AL9 57399563 IC50 = 1310 nM T47941 C7BSY8 57401314 IC50 = 11800 nM T47941 C3QEI9 57401315 IC50 = 3720 nM T47941 COZ7Q8 57401317 IC50 = 2300 nM T47941 CLP9Y6 58607138 IC50 = 3500 nM T47941 CNS12C 59108012 IC50 = 26 nM T47941 C5JZX9 59108013 IC50 = 16 nM T47941 COID58 59108014 IC50 = 18 nM T47941 CAH89G 59108016 IC50 = 12 nM T47941 C1D3RC 59108019 IC50 = 116 nM T47941 CR8W7X 59108022 IC50 = 19 nM T47941 CC57KS 59108026 IC50 = 15 nM T47941 C8DE0Y 59108030 IC50 = 82 nM T47941 CHW15Y 59108031 IC50 = 13 nM T47941 CXP2W3 59108038 IC50 = 54 nM T47941 C3PNK1 59108040 IC50 = 414 nM T47941 CM57VQ 59108041 IC50 = 13 nM T47941 CLN4V3 59108042 IC50 = 28 nM T47941 CX9Z0D 59108044 IC50 = 29 nM T47941 C7PB1U 59321218 IC50 = 4410 nM T47941 CS32XI 59321284 IC50 > 10000 nM T47941 C23WQA 59321310 IC50 > 10000 nM T47941 CZ6C9L 59321318 IC50 > 10001 nM T47941 C1OHZ0 59321339 IC50 > 5000 nM T47941 C7W6BL 60096091 IC50 = 40 nM T47941 C0AFM6 60150358 IC50 = 1910 nM T47941 C6C8RD 66802145 IC50 = 1190 nM T47941 C3KZV7 67494616 IC50 = 1.06 nM T47941 CRIB86 67494620 IC50 = 1.74 nM T47941 CQ3RB9 67494749 IC50 = 4.09 nM T47941 C4J0MF 67863859 IC50 = 20000 nM T47941 CTJ46X 68594477 IC50 > 1000 nM T47941 C8E0XY 68596001 IC50 = 7720 nM T47941 CJ80VI 68596013 IC50 > 10000 nM T47941 CL2H4T 68596452 IC50 > 10000 nM T47941 C93IHS 68596628 IC50 > 10000 nM T47941 CDZ01B 68596639 IC50 > 1000 nM T47941 C1CD9S 68596902 IC50 = 2680 nM T47941 C7PCW0 68597211 IC50 > 1000 nM T47941 CGJB21 68597401 IC50 = 2460 nM T47941 CHK4S0 68597804 IC50 > 10000 nM T47941 C10TGO 68598825 IC50 > 10000 nM T47941 CBP39M 69158736 IC50 = 0.54 nM T47941 CFT3V7 69202515 IC50 = 2400 nM T47941 CC2FG8 69202601 IC50 = 190 nM T47941 COD7R8 69202629 IC50 = 1500 nM T47941 CLHY34 69202696 IC50 = 91 nM T47941 C37HWR 69203016 IC50 = 400 nM T47941 CRP57M 69203166 IC50 = 1800 nM T47941 C3L2KZ 69203269 IC50 > 10000 nM T47941 C5U0FL 69203345 IC50 = 70 nM T47941 COYD87 69203662 IC50 = 140 nM T47941 C7DBC3 69203761 IC50 = 70 nM T47941 C7L2CF 69204029 IC50 = 82 nM T47941 CK3W4E 69204109 IC50 = 3800 nM T47941 CQDT42 69204165 IC50 = 9800 nM T47941 C87NYL 69204282 IC50 = 47 nM T47941 CO60DQ 69204734 IC50 > 10000 nM T47941 CZ89DA 69204736 IC50 = 2000 nM T47941 CS8X9U 69204757 IC50 = 590 nM T47941 C4IZV7 69204803 IC50 = 1300 nM T47941 C3SQI5 69205015 IC50 = 160 nM T47941 CJ52PI 69205027 IC50 = 54 nM T47941 C30UWK 69205046 IC50 = 1900 nM T47941 C0LX2D 69205197 IC50 > 10000 nM T47941 C9MAO5 69205299 IC50 = 3400 nM T47941 C9RY7G 70030919 IC50 = 80 nM T47941 C9BZ8S 70327970 IC50 = 6700 nM T47941 CCN10Q 70662473 IC50 = 0.04 nM T47941 CMD97R 70662578 IC50 = 0.03 nM T47941 CCRS17 70662614 IC50 = 0.41 nM T47941 C5E3JU 70662627 IC50 = 0.12 nM T47941 C82KWY 70680958 IC50 > 10000 nM T47941 CHD8J3 70680959 IC50 = 110 nM T47941 CB31MR 70680960 IC50 = 150 nM T47941 C70QGU 70680962 IC50 = 49 nM T47941 CP21CH 70680964 IC50 = 120 nM T47941 C3EUQ5 70683081 IC50 = 41 nM T47941 C2VG5U 70683082 IC50 = 120 nM T47941 C87JWQ 70683664 IC50 = 2300 nM T47941 C0NFE8 70685170 IC50 = 3600 nM T47941 CM3OP8 70686796 IC50 > 10000 nM T47941 CHBT91 70686797 IC50 > 1000 nM T47941 C4S8KW 70687328 IC50 > 10000 nM T47941 C2O4LX 70689382 IC50 > 10000 nM T47941 CM9QO6 70689383 IC50 = 69 nM T47941 CC5BW9 70691464 IC50 > 10000 nM T47941 CWH57Q 70691484 IC50 = 200 nM T47941 CNJ31P 70695703 IC50 = 52 nM T47941 CC43LF 71074083 IC50 = 289 nM T47941 CG75MJ 71092687 IC50 = 9.44 nM T47941 CR9UP6 71624530 IC50 = 76 nM T47941 C2YCS7 71624531 IC50 = 538 nM T47941 C40NTG 71624532 IC50 = 48 nM T47941 C8RDG9 71624638 IC50 = 10800 nM T47941 C7LFJ0 71624639 IC50 = 365 nM T47941 C03GMI 71624640 IC50 = 1390 nM T47941 CJA8Q5 72713752 IC50 = 23000 nM T47941 C15JYH 73346459 IC50 = 10 nM T47941 CS5XE8 73353458 IC50 = 1.2 nM T47941 C56RIA 73354963 IC50 = 31 nM T47941 CE6OG5 73357099 IC50 = 0.6 nM T47941 C7PVY5 76310476 IC50 = 0.04 nM T47941 C5Z0FC 76310477 IC50 = 4.9 nM T47941 CO8M7V 76314125 IC50 = 1.34 nM T47941 C0Z5DF 76314126 IC50 = 0.22 nM T47941 C7U0VG 76314127 IC50 = 0.16 nM T47941 CNM4F5 76314128 IC50 = 1.85 nM T47941 CD0Z5I 76314129 IC50 = 0.69 nM T47941 CT7RP4 76314130 IC50 = 0.06 nM T47941 C6YKJ4 76314131 IC50 = 0.73 nM T47941 C43UJW 76316861 IC50 = 209.89 nM T47941 CQTO65 76317701 IC50 = 0.2 nM T47941 CYB57F 76317702 IC50 = 0.13 nM T47941 C6R9VE 76317703 IC50 = 0.26 nM T47941 CV8HN6 76317704 IC50 = 0.32 nM T47941 CM4QX0 76317705 IC50 = 0.13 nM T47941 CM9JI6 76321410 IC50 = 0.072 nM T47941 CP0R2W 76321411 IC50 = 0.96 nM T47941 CAZ2C7 76321412 IC50 = 0.18 nM T47941 C0YE2K 76321413 IC50 = 6.83 nM T47941 CN8J7U 76321414 IC50 = 0.07 nM T47941 CNI56P 76325003 IC50 = 0.38 nM T47941 C3HCL5 76325004 IC50 = 0.56 nM T47941 C7OZ9L 76325005 IC50 = 0.06 nM T47941 C16FSI 76325006 IC50 = 0.21 nM T47941 CEUZ92 76325007 IC50 = 0.04 nM T47941 C0EHU7 76325008 IC50 = 0.3 nM T47941 CFN6O9 76325009 IC50 = 0.4 nM T47941 CY45DS 76328577 IC50 = 2.43 nM T47941 CGIY78 76328578 IC50 = 0.1 nM T47941 CU8PB9 76328579 IC50 = 0.75 nM T47941 CM3Y2Q 76328580 IC50 = 0.03 nM T47941 CQ70JV 76328581 IC50 = 0.31 nM T47941 CM7O9S 76328582 IC50 = 0.89 nM T47941 CDZ6P9 76328583 IC50 = 0.04 nM T47941 CJZA18 76332237 IC50 = 3.45 nM T47941 CNJ58D 76332255 IC50 = 44 nM T47941 CW0ME9 76332256 IC50 = 1.9 nM T47941 CCF8B4 76332257 IC50 = 0.21 nM T47941 C9KA7F 76332258 IC50 = 0.08 nM T47941 C0Q9KW 76335878 IC50 = 1.18 nM T47941 C9P8EG 76335892 IC50 = 1.14 nM T47941 C3Y9GR 76335893 IC50 = 0.41 nM T47941 C2DI1C 76335894 IC50 = 0.14 nM T47941 CFR95P 76335895 IC50 = 0.25 nM T47941 C1GW2E 76335896 IC50 = 0.09 nM T47941 CKWR98 76335897 IC50 = 0.21 nM T47941 C4DQ1K 76335898 IC50 = 0.15 nM T47941 CF03DW 90168772 IC50 = 8400 nM T47941 CM6J9K 90168778 IC50 > 20000 nM T47941 CPN65E 90643787 IC50 = 30000 nM T47941 C0E7YS 90662965 IC50 = 9100 nM T47941 CDWL85 90662966 IC50 = 80000 nM T47941 CKES87 90662967 IC50 = 330000 nM T47941 CQ1C3L 90662968 IC50 = 50000 nM T47941 C89MGW 90662969 IC50 = 53000 nM T47941 CZ04FV 90662970 IC50 = 56000 nM T47941 C2TUS1 90662971 IC50 = 37000 nM T47941 C7O5BK 90662972 IC50 = 20000 nM T47941 C3NDF5 90662973 IC50 = 120000 nM T47941 CXW84Y 90662974 IC50 = 17000 nM T47941 C8V2UA 90662975 IC50 = 61000 nM T47941 CFAD54 90662977 IC50 = 3600 nM T47941 CMI17B 90662978 IC50 = 2000 nM T47941 C1UFZ9 90662980 IC50 = 5600 nM T47941 CJG4R7 90662983 IC50 = 1200 nM T47941 CK9ZU1 90662984 IC50 = 80000 nM T47941 CY2B9N 90662985 IC50 = 11000 nM T47941 CD26JN 90662986 IC50 = 33000 nM T47941 C4FO8S 90662987 IC50 = 19000 nM T47941 CE61CW 90662988 IC50 = 11000 nM T47941 CWZ19U 90662989 IC50 = 30000 nM T47941 CV4Z3Y 90662990 IC50 = 40000 nM T47941 CCZ63K 90662992 IC50 = 3500 nM T47941 C20TSL 90662993 IC50 = 53000 nM T47941 C6CF8Z 90662994 IC50 = 25000 nM T47941 C6X4RI 90662995 IC50 = 29000 nM T47941 CPO7B4 90662996 IC50 = 290000 nM T47941 C05TAX 90662999 IC50 = 3600 nM T47941 CMF29Q 90663000 IC50 = 13000 nM T47941 CQ90OV 90663001 IC50 = 27000 nM T47941 C6IO4U 90663002 IC50 = 18000 nM T47941 CK3C4M 90663003 IC50 = 170000 nM T47941 CJG7B9 90663004 IC50 = 13000 nM T47941 C6D7XB 90663005 IC50 = 33000 nM T47941 CFB27O 90663006 IC50 = 100000 nM T47941 C8LOA4 90663007 IC50 = 15000 nM T47941 CAM63V 90663008 IC50 = 7700 nM T47941 C62DWN 90663009 IC50 = 33000 nM T47941 CF1MP2 90665863 IC50 = 372 nM T47941 C1XYI5 90665864 IC50 = 362 nM T47941 C56EKX 90665865 IC50 = 1000 nM T47941 CMP05T 90665866 IC50 = 4700 nM T47941 C4VO0P 90665867 IC50 = 84 nM T47941 CXB56U 90665868 IC50 = 250 nM T47941 C85WCM 90665869 IC50 = 10000 nM T47941 C97KAF 90665870 IC50 = 10000 nM T47941 C6YGD7 90665871 IC50 = 1500 nM T47941 C7SJZ2 90665872 IC50 = 10000 nM T47941 CO3VQ5 90665873 IC50 = 10000 nM T47941 C0B7FJ 90665874 IC50 = 29 nM T47941 CVYK24 118556943 IC50 > 50000 nM T47941 CNGQ19 122179477 IC50 = 5650 nM T47941 CS80MH 122193673 IC50 = 960 nM T47941 CJ7OL5 122193674 IC50 > 100000 nM T47941 C8CJU5 122193675 IC50 = 910 nM T47941 CA60UO 122193676 IC50 > 100000 nM T47941 CAT6J0 122193677 IC50 = 18300 nM T47941 CJ35RG 122193678 IC50 = 11100 nM T47941 CS6M9C 122193679 IC50 = 1100 nM T47941 CE31KJ 122193752 IC50 > 100000 nM T47941 CZB16W 122193753 IC50 = 2200 nM T47941 CQV4W1 122193754 IC50 = 410 nM T47941 C2B4LP 122193755 IC50 > 100000 nM T47941 CL3KD8 122193756 IC50 = 2100 nM T47941 C5DQP9 122193757 IC50 = 12400 nM T47941 C4MZ7H 122193758 IC50 = 6900 nM T47941 COX7E3 122510453 IC50 = 11000 nM T47941 C4AN7Y 127028460 IC50 = 0.55 nM T47941 C31TJD 127028787 IC50 = 1.6 nM T47941 CSY7W4 127029367 IC50 = 0.32 nM T47941 CL8ZE4 127037893 IC50 > 10000 nM T47941 C2A3TY 127038253 IC50 = 5400 nM T47941 C86UVX 127038665 IC50 = 1820 nM T47941 CUA14O 127038666 IC50 = 1500 nM T47941 CY2JI6 127039005 IC50 = 243 nM T47941 C3LWF7 127039006 IC50 = 5600 nM T47941 CTLJ59 127039007 IC50 = 629 nM T47941 C8WQ5K 127039011 IC50 = 130 nM T47941 CSY34W 127039587 IC50 > 10000 nM T47941 CW59OX 127039663 IC50 = 270 nM T47941 CQD37E 127040004 IC50 = 507 nM T47941 C8QM7X 127040005 IC50 = 480 nM T47941 CC71SR 127040006 IC50 = 8 nM T47941 C7V8RC 127040007 IC50 = 5 nM T47941 CI6J9N 127041241 IC50 > 10000 nM T47941 CCNA62 127041543 IC50 > 10000 nM T47941 C1QMI8 135401477 IC50 > 500 nM T47941 C8IUY3 135406430 IC50 = 31000 nM T47941 C17YXR 135406983 IC50 > 500 nM T47941 CJG80M 135412716 IC50 = 2000 nM T47941 C0GQR4 135413516 IC50 = 4000 nM T47941 CMG81E 135434015 IC50 = 6 nM T47941 CK96IT 135436358 IC50 = 600 nM T47941 C94RVJ 135438569 IC50 > 500 nM T47941 CZJY69 135442775 IC50 > 100000 nM T47941 CR6B9J 135456675 IC50 > 100000 nM T47941 CDQJ34 135526598 IC50 = 3100 nM T47941 CP71WA 135528334 IC50 > 100000 nM T47941 C8E3OA 135531470 IC50 > 100000 nM T47941 C4ASW0 135544141 IC50 > 500 nM T47941 C9IJK1 135566935 IC50 = 21200 nM T47941 CJCO05 135750249 IC50 > 20000000 nM T47941 C7H9YC 135750250 IC50 = 8400000 nM T47941 C3LA1D 135750251 IC50 > 20000000 nM T47941 CGJ5E8 135750252 IC50 > 20000000 nM T47941 C62WTU 135750253 IC50 > 20000000 nM T47941 CPU1J3 135750254 IC50 = 159000 nM T47941 C1RK8U 135815296 Ki = 191 nM T47941 C6OU3Z 136034782 IC50 > 500 nM T47941 CECL38 136035345 IC50 = 121000 nM T47941 CW7G2B 136042252 IC50 = 850 nM T47941 C0F6ZG 136058110 IC50 = 6.1 nM T47941 C6N1PA 136058113 IC50 = 5 nM T47941 C6WH2S 136078534 IC50 > 500 nM T47941 CRP24A 136087045 IC50 = 1400 nM T47941 C7SUX4 136087050 IC50 = 13600 nM T47941 C8UF7G 136087052 IC50 = 15700 nM T47941 C4SG1A 136099782 Ki = 436 nM T47941 C2VO1H 136132220 Ki = 35 nM T47941 C8PG9Q 136132221 Ki = 38 nM T47941 CUI4W9 136132222 Ki = 9.3 nM T47941 CST26Q 136132223 Ki = 60 nM T47941 CQ27TM 136132224 Ki = 1210 nM T47941 CMIY85 136132225 Ki = 25 nM T47941 C7J3IT 136132226 Ki = 91.7 nM T47941 CT3IC8 136132227 Ki = 1470 nM T47941 CYM29K 136132228 Ki = 30.3 nM T47941 CEM5N1 136132229 Ki = 5230 nM T47941 C4V5AD 136132230 Ki = 44 nM T47941 CJC0X9 136132231 Ki = 204 nM T47941 COA9T2 136132232 Ki = 22.6 nM T47941 CQ50CG 136132233 Ki = 23.5 nM T47941 CY50JV 136132234 Ki = 19.7 nM T47941 C28IYL 136132235 Ki = 49 nM T47941 CHW75A 136132236 Ki = 26 nM T47941 C9GA2W 136132237 Ki = 58 nM T47941 C39MDZ 136132238 Ki = 15 nM T47941 CW3FM6 136132239 Ki = 25.3 nM T47941 C5XBZ6 136132240 Ki = 53.3 nM T47941 CU8RC1 136132241 Ki = 27 nM T47941 C5NVZ9 136132242 Ki = 45.3 nM T47941 CF31SZ 136132243 Ki = 83.3 nM T47941 CQW7T0 136197286 IC50 > 10000 nM T47941 C2QLX3 138393292 IC50 = 650 nM T47941 CU98MJ 139267730 IC50 = 5830 nM T47941 CMX2Y1 139267731 IC50 = 2730 nM T47941 CVAM65 139399322 IC50 = 2580 nM T47941 CUN3G2 139399340 IC50 = 2710 nM T47941 C87OQT 139399398 IC50 = 2160 nM T47941 C2DA1W 155561694 IC50 > 500000 nM T47941 CQ2R0W 155568588 IC50 > 500000 nM T47941 D00JBC 12905389 Ki = 19100 nM T47941 D00TQR 86344 Ki = 10600 nM T47941 D01RUN 448055 IC50 = 50.12 nM T47941 D02FZD 158758 IC50 = 1100 nM T47941 D02ZPV 10125445 IC50 = 630 nM T47941 D03KKK 169317 Ki = 26100 nM T47941 D04WBU 12905388 Ki = 25000 nM T47941 D05ZUX 44207909 Ki >= 1000 nM T47941 D0A2WH 14969715 Ki = 71100 nM T47941 D0DL6J 9843744 IC50 = 270 nM T47941 D0F1AS 80220 Ki = 163000 nM T47941 D0I6XA 149784 Ki > 200000 nM T47941 D0JD4C 9853498 IC50 = 0.16 nM T47941 D0KD6S 44278378 IC50 = 2200 nM T47941 D0LD0X 128525 Ki = 49300 nM T47941 D0LZ5R 5368 IC50 = 67000 nM T47941 D0M5NU 161733 IC50 = 130000 nM T47941 D0O3BL 19700663 IC50 = 56 nM T47941 D0S4JI 20262 IC50 = 160000 nM T47941 D0T2RY 9948320 Ki >= 1000 nM T47941 D0V4WB 149790 IC50 = 1700 nM T47941 D0V5BX 68765 IC50 = 50 nM T47941 D0W7WV 11039077 IC50 = 5 nM T00895 D01XYJ 35370 IC50 > 150000 nM T00895 D03KKR 3547 IC50 = 3000 nM T00895 D09DHT 27924 Ki = 0.45 nM T00895 D0E3TC 44259 IC50 = 0.6 nM T00895 D0I6VU 176167 IC50 = 300 nM T00895 D0LF1U 5287969 IC50 = 480 nM T00895 D0MS3Z 16725726 IC50 = 21 nM T00895 D0R9YR 64971 IC50 > 150000 nM T00895 D0W3LI 153999 IC50 = 600 nM T00895 D03BNU 59604787 IC50 > 10000 nM T00895 D0WS1V 448991 IC50 > 100000 nM T00895 D0R2TM 5287736 IC50 = 10 nM T00895 C8OI7N 2290 IC50 = 38 nM T00895 C95GCZ 3568 IC50 = 108 nM T00895 CJ17AM 4877 IC50 = 21 nM T00895 C91OFE 64980 IC50 > 150000 nM T00895 C5KW4H 72311 IC50 = 24 nM T00895 CG2P1X 159320 Ki = 1 nM T00895 C8PU1O 188534 Ki = 0.47 nM T00895 C75EDQ 644355 IC50 = 30000 nM T00895 C5HPF3 644356 IC50 > 100000 nM T00895 C6DLK3 644364 IC50 = 39000 nM T00895 CLBZ39 2272071 IC50 = 28500 nM T00895 C5M4LH 3167689 IC50 = 25500 nM T00895 CNW2D8 3207458 IC50 = 11200 nM T00895 CTID76 5282335 IC50 = 5600 nM T00895 CLA43B 5327919 IC50 = 280 nM T00895 CPDC54 5327920 IC50 = 1800 nM T00895 CCB9G3 5327921 IC50 = 10 nM T00895 CRTQ98 5327922 IC50 = 50 nM T00895 CP20NQ 5327923 IC50 = 30 nM T00895 C98CNM 5327943 IC50 = 13000 nM T00895 C61URB 5327944 IC50 = 50 nM T00895 CWUY53 5327945 IC50 = 15000 nM T00895 CQ54BE 5327946 IC50 = 320 nM T00895 CIB3P0 5327947 IC50 = 2300 nM T00895 CVG0A1 5327948 IC50 = 460 nM T00895 C8M3PD 5327949 IC50 > 50000 nM T00895 CA25BM 5327950 IC50 > 50000 nM T00895 COP0Q2 5327951 IC50 = 30000 nM T00895 CB47VN 5327952 IC50 = 4100 nM T00895 CPO51K 5327953 IC50 = 280 nM T00895 CI6AY9 5327954 IC50 > 50000 nM T00895 C1Q0PM 5327955 IC50 > 50000 nM T00895 CXA23M 5327956 IC50 = 47000 nM T00895 CH73DT 5327957 IC50 = 30000 nM T00895 CTI6K8 5327963 IC50 = 13000 nM T00895 CAO1N9 5327979 IC50 = 370 nM T00895 CMP3X8 5327994 IC50 = 310 nM T00895 C4DG8Y 5327995 IC50 = 2000 nM T00895 CDL0S2 5327996 IC50 > 50000 nM T00895 CC43JH 5327997 IC50 = 32000 nM T00895 CKS8M6 5327998 IC50 = 2000 nM T00895 CQ7OZ6 5327999 IC50 = 3800 nM T00895 CQWO93 5328000 IC50 = 4700 nM T00895 CU73IX 5328002 IC50 = 170 nM T00895 CTVP40 5328003 IC50 = 1300 nM T00895 CBSP34 5328004 IC50 = 3700 nM T00895 CS78OD 5328005 IC50 = 3200 nM T00895 CO9YQ6 5328006 IC50 = 25000 nM T00895 CVX2L3 5328007 IC50 = 34 nM T00895 CPD1U9 5328008 IC50 = 130 nM T00895 C3X6QJ 5328012 IC50 = 660 nM T00895 CZO4E1 5328013 IC50 = 13000 nM T00895 C9NBG7 5330546 IC50 > 100000 nM T00895 C2RA4O 5352033 Ki = 0.63 nM T00895 CW1ZY2 6520576 Ki = 1.03 nM T00895 CG17TN 6914611 IC50 = 6100 nM T00895 C0IK9O 9543716 EC50 = 14270 nM T00895 C4PA5X 9800852 Ki = 469 nM T00895 C8J1OL 9826373 IC50 = 900 nM T00895 CP17TY 9847089 IC50 = 10 nM T00895 CCJK12 9865633 Ki = 40 nM T00895 C20NKA 9889351 IC50 = 400 nM T00895 C9O3XQ 9901617 IC50 = 335 nM T00895 CP5NJ3 9952970 Ki = 13.1 nM T00895 CV34AB 9958125 IC50 = 4000 nM T00895 C2W3AV 9995236 IC50 = 4000 nM T00895 CY65CO 10030073 IC50 = 300 nM T00895 C2UGV9 10030483 IC50 = 16000 nM T00895 CT6BJ7 10099352 IC50 > 150000 nM T00895 CG7JO8 10099482 IC50 = 5900 nM T00895 C93LPQ 10099652 IC50 = 170 nM T00895 CEF8U5 10117705 IC50 = 250 nM T00895 C2O7ZH 10137972 IC50 = 4.3 nM T00895 C91BQM 10147482 IC50 = 1020 nM T00895 CGOT91 10207821 IC50 = 75 nM T00895 CI8MW4 10216627 IC50 > 5000 nM T00895 C8W2HS 10224497 Ki = 121.3 nM T00895 C3VK7T 10229967 IC50 = 170 nM T00895 C7SFI1 10296883 IC50 = 6.2 nM T00895 CMK32F 10300534 IC50 > 150000 nM T00895 CFU38G 10363814 Ki = 411 nM T00895 CEH41V 10392789 IC50 = 30 nM T00895 C3RBY8 10395226 Ki = 17.9 nM T00895 CDR7X8 10415328 IC50 > 150000 nM T00895 CQXJ51 10425978 Ki = 41.5 nM T00895 C36QRS 10453829 Ki = 540 nM T00895 C10PAC 10460251 IC50 = 160 nM T00895 C25LDK 10460643 IC50 > 50000 nM T00895 C1VI3E 10477747 IC50 = 285 nM T00895 CMA4J8 10479260 Ki = 228 nM T00895 C70SUP 10482065 IC50 > 150000 nM T00895 CX7S8N 10482293 IC50 = 10 nM T00895 C76QGP 10506540 IC50 = 150 nM T00895 CSR8Y5 10527068 IC50 > 5000 nM T00895 CDNP37 10530708 IC50 = 270 nM T00895 C5EYJ3 10554684 IC50 = 1000 nM T00895 C71UIS 10555532 IC50 = 45000 nM T00895 CZ8UA9 10650891 IC50 > 5000 nM T00895 CJOU71 10671412 IC50 = 1100 nM T00895 CM5B6A 10673286 IC50 > 5000 nM T00895 CN9I6T 10768377 IC50 > 5000 nM T00895 CL8VH3 10768554 IC50 = 57000 nM T00895 C5YMK8 10769011 IC50 = 30 nM T00895 C7HPA0 10864309 IC50 = 6000 nM T00895 C1DRE5 10884145 IC50 = 30 ug.mL-1 T00895 C2G5CU 10894726 Ki = 262 nM T00895 C1L4ZC 10940039 IC50 = 9400 nM T00895 CR47CD 11025838 Ki = 83 nM T00895 C67CSJ 11201611 IC50 = 18 nM T00895 C3ROM0 11247414 IC50 = 182 nM T00895 CRZ38O 11315034 IC50 = 225 nM T00895 C4ON7Z 11362429 IC50 = 4.3 nM T00895 C8DNQ2 11453012 IC50 = 1000 nM T00895 C3KAC4 11538477 IC50 > 316 nM T00895 C1CD2N 11547825 IC50 = 251 nM T00895 C9OV5S 11561609 IC50 = 73 nM T00895 CACS26 11561968 Ki > 10000 nM T00895 CD7PF5 11574473 IC50 > 316 nM T00895 CA9XJ2 11604381 IC50 = 30 nM T00895 CI9HQ2 11624816 IC50 > 316 nM T00895 CQ5S3G 11639520 IC50 > 316 nM T00895 CU0E8O 11690457 Ki = 690 nM T00895 CB0AP2 11705863 Ki > 10000 nM T00895 CCX53Q 11729563 IC50 = 50 nM T00895 C17SIL 11756581 IC50 > 150000 nM T00895 CM10YB 11799388 IC50 = 3800 nM T00895 CTN96I 11851810 IC50 = 0.9 nM T00895 CA05OS 11972484 IC50 = 3600 nM T00895 CQ39BY 12115602 IC50 = 5.5 nM T00895 C2BX8F 15297223 IC50 = 340 nM T00895 CE04YW 15297224 IC50 > 50000 nM T00895 C7N6CQ 15604547 IC50 = 8300 nM T00895 C9TU1O 16046126 IC50 > 1000 nM T00895 CZF23I 16124479 IC50 = 398.11 nM T00895 CC24KI 16667248 IC50 = 610 nM T00895 CFAR38 17814740 IC50 > 10000 nM T00895 C9AVK0 21113469 IC50 > 315 nM T00895 CS15LY 21672114 Ki = 1.3 nM T00895 CZ0X8J 22592015 IC50 > 315 nM T00895 CVR9K4 22907281 IC50 = 390 nM T00895 C0HRM6 22911602 IC50 = 400 nM T00895 CUN67H 23366085 IC50 = 14000 nM T00895 CLG9Z8 23366090 IC50 = 27000 nM T00895 CW6OB1 23627212 IC50 = 2.5 nM T00895 CKYB29 23644745 IC50 = 970 nM T00895 C2JTA3 23647573 IC50 = 8900 nM T00895 CK73JS 24742033 Ki = 29 nM T00895 CK60ZM 24758992 IC50 > 8000 nM T00895 C2UOE0 24766030 IC50 = 3000 nM T00895 CJUK39 24770517 IC50 = 2330 nM T00895 CM28WD 24825721 IC50 = 54 nM T00895 CZ2PQ6 24863113 IC50 > 8000 nM T00895 CBYM61 24863535 IC50 > 8000 nM T00895 CSW5V3 24865437 IC50 = 39 nM T00895 CS3Q8B 24995659 Ki = 17 nM T00895 C1ONA4 24996161 IC50 = 18 nM T00895 CXJ2H9 25052849 Ki = 2.57 nM T00895 CQNK94 25053046 Ki = 18.2 nM T00895 C0G1KQ 25053118 Ki = 18.3 nM T00895 C0OI9H 25053465 Ki = 39.4 nM T00895 C0W2LR 25053469 Ki = 13.4 nM T00895 C6AQE3 25053483 Ki = 380 nM T00895 CX7A0N 25053598 Ki = 21.1 nM T00895 CSW45A 25053658 Ki = 220 nM T00895 C53ZIQ 25053780 Ki = 328 nM T00895 CAED20 25053782 Ki = 199 nM T00895 CZO27W 25054032 IC50 > 5000 nM T00895 CN2G3K 25054307 IC50 > 5000 nM T00895 C7IZ6K 25055317 IC50 > 5000 nM T00895 CFHO90 25056112 IC50 > 5000 nM T00895 CU8X0H 25056370 IC50 > 5000 nM T00895 CV15HY 25056371 IC50 > 5000 nM T00895 C76LFY 25056889 IC50 > 5000 nM T00895 CH6AU8 25057408 IC50 > 5000 nM T00895 C0B7RT 25057409 IC50 > 5000 nM T00895 C3AT0H 25057667 IC50 > 5000 nM T00895 CH7YC4 25057933 IC50 > 5000 nM T00895 C6P1CX 25066843 IC50 = 17 nM T00895 CDO3X2 25113021 IC50 = 79 nM T00895 CBI73N 25113026 IC50 = 44 nM T00895 C1R0JL 25113028 IC50 = 13 nM T00895 C4KL8Q 25113038 IC50 = 62 nM T00895 CV58WZ 25113039 IC50 = 403 nM T00895 C8KI1Z 25113050 IC50 = 802 nM T00895 CD5Z8U 44139091 Ki = 78.7 nM T00895 CAI56R 44139212 Ki = 147 nM T00895 CNX5R1 44139336 Ki = 31.9 nM T00895 CRD90G 44139337 Ki = 8.3 nM T00895 C4UMB7 44158300 Ki = 25 nM T00895 C4G5DI 44158301 Ki = 820 nM T00895 CLW80F 44160269 IC50 = 14 nM T00895 CYE36B 44241613 IC50 > 40000 nM T00895 C6LG5T 44241614 IC50 > 40000 nM T00895 CIX8V2 44251637 IC50 = 16 nM T00895 C5QFX6 44263382 IC50 = 29 nM T00895 C8RQU2 44263383 IC50 = 59 nM T00895 CZG81D 44263384 IC50 = 19 nM T00895 C6YRP1 44263385 IC50 = 1825 nM T00895 CQ13XB 44291629 Ki = 489.6 nM T00895 CERT91 44291669 Ki = 55 nM T00895 C1FZ6B 44294270 IC50 = 4500 nM T00895 C6A9FK 44294365 IC50 = 10 nM T00895 C4HS3C 44294447 IC50 = 120 nM T00895 CFZ31C 44294493 IC50 = 240 nM T00895 C54GFD 44294623 IC50 = 20 nM T00895 CG89DS 44294661 IC50 = 4000 nM T00895 CSHC96 44297347 IC50 = 2900 nM T00895 CYF8O6 44297594 IC50 = 640 nM T00895 CG1Z2B 44303442 IC50 = 50 nM T00895 CNJ63O 44303517 IC50 = 80 nM T00895 C8RJN7 44303745 IC50 = 670 nM T00895 CTM59P 44308069 IC50 = 10 nM T00895 CJ4WB9 44308383 IC50 = 150 nM T00895 C1N6SL 44308409 IC50 = 16000 nM T00895 CO83HF 44308467 IC50 = 5900 nM T00895 CYTA85 44308468 IC50 = 45000 nM T00895 C3M4UP 44308469 IC50 = 280 nM T00895 CY4K5F 44308490 IC50 = 49 nM T00895 C7AG9Y 44308609 IC50 = 160 nM T00895 CYN34A 44308610 IC50 = 30 nM T00895 C79WUE 44308611 IC50 = 30 nM T00895 CS63CK 44308612 IC50 = 260 nM T00895 C47BNR 44310732 IC50 = 10 nM T00895 C2ACB1 44310758 IC50 = 50 nM T00895 CXVB19 44310795 IC50 = 40000 nM T00895 CD8OF2 44311036 IC50 = 15 nM T00895 C13TNU 44315122 IC50 = 250 nM T00895 C3YN1R 44315123 IC50 = 3700 nM T00895 CPJ57U 44315124 IC50 = 50 nM T00895 C9HA8T 44315171 IC50 = 100 nM T00895 C2T3VN 44315184 IC50 = 3600 nM T00895 C3SP0H 44315423 IC50 = 3600 nM T00895 C8OAE9 44315457 IC50 = 1300 nM T00895 C3JS6X 44315503 IC50 = 30 nM T00895 CEZ68T 44315545 IC50 = 4800 nM T00895 C73MZU 44322457 IC50 = 6700 nM T00895 C2C3MV 44322458 IC50 = 2100 nM T00895 CA4R8N 44322474 IC50 = 3300 nM T00895 C2WUL9 44322520 IC50 = 8000 nM T00895 C3DY4L 44322570 IC50 = 310 nM T00895 C3UMR9 44322571 IC50 = 410 nM T00895 CE0QG3 44322667 IC50 = 4700 nM T00895 C31QSE 44322668 IC50 = 3800 nM T00895 CIB64S 44322669 IC50 = 4600 nM T00895 C42OZF 44322670 IC50 = 16000 nM T00895 CPL9E5 44322671 IC50 > 5000 nM T00895 C17GFI 44322684 IC50 = 39000 nM T00895 CG2SL8 44322685 IC50 = 370 nM T00895 CU8CK7 44322686 IC50 = 97000 nM T00895 COCR18 44322713 IC50 = 3500 nM T00895 C6DHT8 44322714 IC50 = 10000 nM T00895 CK7CJ9 44322718 IC50 = 30000 nM T00895 C3VA0L 44322719 IC50 = 4300 nM T00895 C6Z9XL 44322720 IC50 > 50000 nM T00895 C8NR7B 44322740 IC50 = 8100 nM T00895 C4X3UE 44322741 IC50 = 47000 nM T00895 C1JY5B 44322762 IC50 = 36000 nM T00895 CGK4V2 44322763 IC50 = 38 nM T00895 CP2X6J 44322771 IC50 = 5000 nM T00895 CA27PF 44322772 IC50 = 830 nM T00895 C4P5HM 44322773 IC50 = 2600 nM T00895 CZ7N8D 44322811 IC50 = 2200 nM T00895 C4J3RI 44322813 IC50 = 2000 nM T00895 CI6R4S 44322889 IC50 > 150000 nM T00895 C48NJC 44322981 IC50 = 300 nM T00895 C6K5TE 44322982 IC50 > 150000 nM T00895 CFMB02 44323003 IC50 > 50000 nM T00895 CF61IT 44334334 IC50 = 80 nM T00895 C3BFI4 44334443 IC50 = 310 nM T00895 CKD2B8 44337790 IC50 > 150000 nM T00895 COJ73E 44355185 Ki = 0.55 nM T00895 CIH03D 44366053 IC50 = 38000 nM T00895 CO28BT 44376126 Ki = 0.58 nM T00895 C8X0WA 44384580 Ki = 515 nM T00895 CC95JU 44385548 IC50 < 1000 nM T00895 CGQ57L 44386180 IC50 = 480 nM T00895 CI0Y5L 44386181 IC50 = 50 nM T00895 C1W6NC 44386587 IC50 = 10 nM T00895 C0PU3I 44386588 IC50 = 310 nM T00895 C3J6ZO 44386589 IC50 = 1900 nM T00895 C4MZI9 44386931 IC50 = 25000 nM T00895 C8B1LV 44394308 IC50 = 3425 nM T00895 C4UR6L 44394355 IC50 = 58 nM T00895 C9CX5A 44394369 IC50 > 10000 nM T00895 CKCW90 44394463 IC50 > 10000 nM T00895 CA7ZI5 44394482 IC50 = 3455 nM T00895 CP9CT3 44394511 IC50 = 3905 nM T00895 CFX48I 44394512 IC50 = 6322 nM T00895 CS83VP 44394536 IC50 = 3456 nM T00895 CIY32A 44394554 IC50 = 5866 nM T00895 C6EZ8Y 44394557 IC50 = 2605 nM T00895 CGXQ92 44425746 Ki = 2.37 nM T00895 COT05F 44450721 IC50 = 39 nM T00895 CY87UN 44456923 Ki = 80.1 nM T00895 CW0T1S 44456924 Ki = 407 nM T00895 CS2CV1 44456938 Ki = 22.5 nM T00895 C5WL1F 44473009 IC50 = 2.5 nM T00895 CEG1S5 44473011 IC50 = 6.5 nM T00895 C46OMR 44473016 IC50 = 8 nM T00895 C0TUS2 44561670 Ki = 41.5 nM T00895 CJY8S0 44570884 IC50 = 95000 nM T00895 C1S8MC 44575685 IC50 > 150000 nM T00895 CSI0U1 44819541 IC50 = 3000 nM T00895 C87FEM 45270051 IC50 > 40000 nM T00895 CU53FK 45273505 IC50 > 40000 nM T00895 CC95PQ 45375865 IC50 = 1.6 nM T00895 CEOQ27 45375866 IC50 = 36 nM T00895 C5S8MA 45485083 IC50 = 7 nM T00895 CW42YX 45487634 IC50 = 12 nM T00895 CQW97N 46846072 IC50 = 2 nM T00895 CXUO70 46890036 IC50 > 8000 nM T00895 CZ2V8R 46890138 IC50 > 8000 nM T00895 CSV5B9 46901859 IC50 = 5 nM T00895 C7YJ2X 46901862 IC50 = 8 nM T00895 CCL6T7 49870878 IC50 = 19952.62 nM T00895 CM42BY 51000510 Ki > 1000000 nM T00895 CHP06V 52948258 Ki = 37 nM T00895 CD4H3S 53354074 Ki = 1 nM T00895 CUY9G2 53473663 IC50 = 72 nM T00895 CGQ7F8 53473746 IC50 = 6.2 nM T00895 CI1ZG3 53473747 IC50 = 2 nM T00895 C67JHW 53473748 IC50 = 3.9 nM T00895 C7EW6O 53473749 IC50 = 16 nM T00895 CPH34R 53473750 IC50 > 316 nM T00895 CWH1D4 53473825 IC50 > 316 nM T00895 CM8K2V 53473826 IC50 = 15.3 nM T00895 C9A8HG 53473827 IC50 > 316 nM T00895 C3A8OT 53473828 IC50 = 334 nM T00895 CLX31Q 53473829 IC50 > 316 nM T00895 C8Y9RE 53473918 IC50 = 9.8 nM T00895 C1XFN0 53473919 IC50 = 32 nM T00895 CN34UO 53473920 IC50 = 19 nM T00895 C2RE5M 53473921 IC50 = 0.7 nM T00895 C9ZUL0 53473922 IC50 = 25 nM T00895 CG6FD5 53474007 IC50 = 11 nM T00895 C0Q7JS 53474008 IC50 = 73 nM T00895 C31WZB 53474009 IC50 = 3.8 nM T00895 CJF1M2 53630890 IC50 = 402 nM T00895 CCM71K 54669828 Ki = 480 nM T00895 CNB76L 56643505 IC50 = 5 nM T00895 CE25GK 57392822 EC50 = 23380 nM T00895 C3GKF9 57969582 Ki = 183 nM T00895 C8W1QC 57969676 Ki = 25 nM T00895 COH41P 58325285 IC50 = 16 nM T00895 CJ6ZT2 59332810 IC50 = 147 nM T00895 COH62U 60097413 IC50 > 10000 nM T00895 C1MR8Q 60097495 IC50 > 1000 nM T00895 CNL04P 60155126 Ki = 17 nM T00895 C56PUM 60155209 Ki = 2 nM T00895 CWTG65 60199327 Ki = 8.08 nM T00895 CV63UL 67240318 IC50 > 10000 nM T00895 CF39DV 68596931 IC50 = 8 nM T00895 C9XLB3 68597337 IC50 = 7 nM T00895 CMQ58W 68597501 IC50 = 81 nM T00895 CEZU83 68611347 IC50 = 120 nM T00895 CJ8G3H 68682755 IC50 > 316 nM T00895 C0HA8V 68783839 IC50 = 82 nM T00895 CJGH31 70285522 IC50 > 1000 nM T00895 CPZ4F6 71451107 IC50 > 1000 nM T00895 C5RKX0 71452928 IC50 = 38 nM T00895 CLZ67D 71456431 IC50 = 929 nM T00895 CS89CL 71456432 IC50 = 24 nM T00895 CPIH21 71460129 IC50 = 47 nM T00895 C69NCX 71461845 IC50 = 877 nM T00895 C9QB5V 71461846 IC50 > 1000 nM T00895 C6O8KG 71461847 IC50 = 133 nM T00895 CU60JG 71718528 IC50 > 50000 nM T00895 CV70GZ 71728100 Ki = 1.3 nM T00895 C2XZW3 72708899 IC50 > 40000 nM T00895 CKN46T 72708901 IC50 > 40000 nM T00895 C7Q0AD 76286479 IC50 = 460 nM T00895 CZF0N7 76287389 IC50 = 140 nM T00895 CS4G0K 86291004 Ki = 14.6 nM T00895 CXPB19 90644017 Ki = 2.17 nM T00895 C6FO1X 90644018 Ki = 11.7 nM T00895 COR0J2 90656209 IC50 = 1020 nM T00895 CF89DA 90664659 IC50 = 5100 nM T00895 C5CKD3 91754690 Ki = 41 nM T00895 C5UTH1 118706399 Ki = 78 nM T00895 CC9F4Q 118706400 Ki = 90 nM T00895 C12BEC 118706401 Ki = 194 nM T00895 C8R2XG 118706402 Ki = 145 nM T00895 C20PIN 118706403 Ki = 119 nM T00895 CVNL09 118706404 Ki = 32 nM T00895 C2LOB4 118706405 Ki = 50 nM T00895 CV4RS5 118706406 Ki = 34 nM T00895 CW03BD 118706407 Ki = 51 nM T00895 CHK86P 118706408 Ki = 30 nM T00895 C74HPT 118706409 Ki = 49 nM T00895 CBDA05 118706410 Ki = 215 nM T00895 C0IRE2 118706411 Ki = 267 nM T00895 CU2RH8 118706412 Ki = 446 nM T00895 C31FCD 118706413 Ki = 26 nM T00895 CLUN23 118706414 Ki = 37 nM T00895 CQKD05 118706415 Ki = 77 nM T00895 CE23GF 118725578 Ki = 12.2 nM T00895 CGJ59M 118725630 Ki = 2.14 nM T00895 C9CQ6J 118725631 Ki = 9.8 nM T00895 CKV3Z1 118725632 Ki = 5.5 nM T00895 CWV1H6 118725633 Ki = 16.3 nM T00895 CS63AL 118725634 Ki = 7.46 nM T00895 CMY94J 118725635 Ki = 19.3 nM T00895 CYRA47 118725636 Ki = 11.4 nM T00895 CWB3J2 118725637 Ki = 1.21 nM T00895 CZI2W3 118725638 Ki = 7.12 nM T00895 CT6S2F 118725639 Ki = 4.79 nM T00895 C64AMW 118725640 Ki = 13.4 nM T00895 C5W3SJ 118725641 Ki = 5.24 nM T00895 CC3NO0 118725642 Ki = 5.06 nM T00895 CF3CU5 118725643 Ki = 4.1 nM T00895 CDH1U2 118725644 Ki = 15.2 nM T00895 C1G5IE 118725645 Ki = 8.3 nM T00895 C5JX1Z 118725646 Ki = 11.5 nM T00895 CRP91U 118725647 Ki = 5.9 nM T00895 C2VQW1 134817176 Ki = 78.9 nM T00895 CSB0M9 135494223 EC50 = 18810 nM T00895 CEK31P 135566415 IC50 > 20000 nM T00895 C1XQY2 135923992 EC50 = 11810 nM T00895 C39NGD 136026545 IC50 > 50000 nM T00895 CC65KF 136042192 EC50 = 16090 nM T00895 C4P5AE 137631716 Ki = 301 nM T00895 C21SUB 137638899 Ki = 119 nM T00895 CHSJ08 137640349 Ki = 55 nM T00895 C12UXT 137640959 IC50 > 316 nM T00895 CH15QZ 137643717 IC50 = 223 nM T00895 C3A9TX 137646224 Ki = 295 nM T00895 CW1TJ7 137649466 Ki = 27.3 nM T00895 CUG6N7 137660315 IC50 = 110 nM T00895 CAS65V 137660703 Ki = 59.6 nM T00895 C4RTS3 137661076 Ki = 131 nM T00895 C6QA5D 137661222 IC50 > 316 nM T00895 C49QOZ 138393053 IC50 = 350 nM T00895 C7ELX9 145949146 Ki = 3408 nM T00895 CZO0S7 145949469 Ki = 6.51 nM T00895 CG1V9D 145949968 Ki = 6.8 nM T00895 CS75PX 145950212 Ki = 8.17 nM T00895 CVY36T 145951556 Ki = 208 nM T00895 CDM0F1 145951838 Ki = 1124 nM T00895 CE1WI4 145951934 Ki = 9.5 nM T00895 CEX16N 145951949 Ki = 12.5 nM T00895 CHB38K 145953902 Ki = 208 nM T00895 C8MCT0 145954310 Ki = 122 nM T00895 CDQU92 145954325 Ki = 6.39 nM T00895 CY0ID9 145954400 Ki > 30000 nM T00895 CKL8B4 145954900 Ki = 780 nM T00895 C4HP0N 145955235 Ki = 130.9 nM T00895 CK9IQ0 145955940 Ki = 19.36 nM T00895 C0G9KP 145956414 Ki = 19.18 nM T00895 CMRB05 145956847 Ki = 73.3 nM T00895 CYD17P 145957502 Ki = 7.87 nM T00895 CS60UE 145957652 Ki = 39.3 nM T00895 CVK9L5 145958383 Ki = 672 nM T00895 C8UQB9 145958537 Ki = 98.2 nM T00895 CHFN64 145958744 Ki = 10.14 nM T00895 CTK58B 145959420 Ki = 103.6 nM T00895 CFWM04 145959424 Ki = 42 nM T00895 CQ7S6Z 145959564 Ki > 30000 nM T00895 C0U5CQ 145961000 Ki = 35.3 nM T00895 C9IY7P 145964008 IC50 = 170 nM T00895 C4ZU2L 145965049 IC50 = 570 nM T00895 CIQ70O 145966247 IC50 = 4200 nM T00895 CPH9E3 145967023 IC50 = 560 nM T00895 C2TMZ3 145967445 IC50 = 45 nM T00895 CXS3W4 145971204 Ki = 7.1 nM T00895 C3PO1Q 145971398 IC50 = 230 nM T00895 C94NTF 145971693 Ki = 60.6 nM T00895 CMXU60 145972550 IC50 = 3300 nM T00895 C98QCL 145974536 Ki = 92.3 nM T00895 C53VBI 145974831 IC50 = 5800 nM T00895 C4FP9E 145975243 IC50 = 530 nM T00895 CMH8Q5 145975400 IC50 = 520 nM T00895 C5V0AH 145977027 IC50 = 3400 nM T00895 C1QY5N 145977386 IC50 = 1100 nM T00895 C2MD1Q 155513187 IC50 > 10000 nM T00895 CZQM57 155554194 IC50 > 10000 nM T00895 D02KPV 37783 Ki = 1.35 nM T00895 D02XHC 448912 IC50 > 100000 nM T00895 D04AXH 11574614 Ki = 510 nM T00895 D05KJY 72326 IC50 > 150000 nM T00895 D06ZCX 10455969 IC50 = 79000 nM T00895 D07ANB 148879 EC50 = 8190 nM T00895 D07OAT 456214 IC50 > 100000 nM T00895 D0H7DQ 6419755 IC50 = 2800 nM T00895 D0K5ZY 105000 Ki = 7.7 nM T00895 D0L8HO 2399 IC50 = 7516 nM T00895 D0N1UU 46871820 IC50 = 1000 nM T00895 D0TO6S 2396 IC50 = 12 nM T00895 D0V0KA 24863112 IC50 > 8000 nM T00895 D0X2DH 17814743 IC50 > 10000 nM T00895 D0XS9E 5330535 IC50 > 30000 nM T46360 D00HPK 47641 Ki = 880 nM T46360 D01AZG 5073 Ki = 4300 nM T46360 D01JUF 5775 IC50 = 549.54 nM T46360 D01XBA 5035 Ki = 38 nM T46360 D01ZSO 4235 Ki > 100 nM T46360 D02KRS 2130 Ki = 20.25 nM T46360 D03HFG 5324346 Ki = 36 nM T46360 D03QGM 5355 IC50 > 10000 nM T46360 D03SKD 5284603 Ki > 10000 nM T46360 D04XPW 446220 Ki = 8830 nM T46360 D06XMU 6013 Ki = 1200 nM T46360 D07BSQ 5994 Ki = 260 nM T46360 D07KSG 2733526 Ki = 35 nM T46360 D08VRO 3822 IC50 = 1 nM T46360 D09OBB 5360696 Ki = 348 nM T46360 D09VBC 2562 Ki = 19.5 nM T46360 D0CT9Y 1548953 Ki = 8 nM T46360 D0D1AL 3559 Ki = 0.2 nM T46360 D0D7TB 9417 Ki = 0.2 nM T46360 D0E1WI 3345 IC50 = 354 nM T46360 D0G8NN 119570 Ki = 4446 nM T46360 D0H6QU 6005 IC50 > 10000 nM T46360 D0H8QL 4020 IC50 = 234.42 nM T46360 D0I0DL 3689 IC50 = 3.9 nM T46360 D0K0TC 68617 Ki = 57 nM T46360 D0L5WM 2157 Ki = 1 nM T46360 D0M8VE 71360 IC50 = 64 nM T46360 D0NS6H 3152 Ki = 14.6 nM T46360 D0P6UB 10836 Ki = 8320 nM T46360 D0R4OM 5566 Ki = 15 nM T46360 D0T8GD 89594 IC50 > 10000 nM T46360 D0TR5X 3386 IC50 = 851.14 nM T46360 D0U2OO 2477 IC50 = 36.31 nM T46360 D0WE3O 5288826 Ki > 10000 nM T46360 D0X3FX 5284596 IC50 > 100000 nM T46360 D0Z1RV 135398737 Ki = 8500 nM T46360 D0Z6ST 2467 Ki = 1290 nM T46360 D00POS 9931976 Ki = 451 nM T46360 D00WLO 3455 IC50 = 43 nM T46360 D0A7KI 3037308 Ki = 490 nM T46360 D0I8FV 5567 Ki = 0.83 nM T46360 D0N1HW 5311200 Ki = 130 nM T46360 D0P1YE 9852175 Ki = 940 nM T46360 D0R8GR 9892540 IC50 = 47 nM T46360 D00KVE 9907323 Ki = 3.162 nM T46360 D0K6NS 6536 Ki = 8 nM T46360 D0H2SE 118607347 Ki = 23 nM T46360 D0N6JH 24968535 Ki = 1437 nM T46360 D0W3TS 41306362 Ki = 3.2 nM T46360 D00EZE 3047810 Ki = 19 nM T46360 D00ZGA 9917021 Ki = 2980 nM T46360 D01KIU 126402 Ki = 46.5 nM T46360 D01PIL 54477 Ki = 55 nM T46360 D01YOC 108046 Ki = 71 nM T46360 D02KLW 180081 IC50 > 10000 nM T46360 D07KYU 9330 Ki > 1000 nM T46360 D07ODD 132891 Ki > 6270 nM T46360 D08AWI 11430856 Ki = 100 nM T46360 D09DRG 9952420 IC50 = 1.3 nM T46360 D0M9GE 53389 IC50 = 450 nM T46360 D0OC3J 5281881 IC50 = 2.239 nM T46360 D0XK2K 9829526 Ki = 17 nM T46360 D0Z4QV 121967 Ki = 10 nM T46360 C5H0QN 1235 Ki = 59.7 nM T46360 C5IOL8 4910 Ki = 17 nM T46360 CW56ZA 5290 Ki = 269 nM T46360 C1WK2E 5417 Ki = 2.5 nM T46360 CE41ZK 7594 IC50 = 397 nM T46360 CP0O8I 9513 Ki = 309 nM T46360 CZC17M 9669 Ki = 36.5 nM T46360 C5VS0H 10098 Ki > 100000 nM T46360 CVW5J9 10220 Ki = 106 nM T46360 CTC8N0 14657 IC50 > 100000 nM T46360 C5EO7I 22648 IC50 = 2200 nM T46360 CM4VK9 33142 Ki = 27.7 nM T46360 CNZD18 36381 Ki = 30.1 nM T46360 C8Y6DE 37461 IC50 = 52.48 nM T46360 CO6M2K 41011 Ki = 3.1 nM T46360 CTF7Z4 50266 Ki = 230 nM T46360 CY2F8T 55445 IC50 = 76 nM T46360 C0RV1Y 60840 IC50 = 2540 nM T46360 C8CZ1E 64600 IC50 = 5 nM T46360 C0LQ7N 65638 Ki = 1 nM T46360 CLY10I 65659 Ki > 100 nM T46360 CDQX62 66270 Ki > 800 nM T46360 C0SKG4 66749 IC50 = 1250 nM T46360 C3WKC6 68835 IC50 = 27200 nM T46360 CZ6G7B 69873 Ki = 1980 nM T46360 CY79XW 72027 Ki = 4 nM T46360 C13JOV 75994 Ki = 10480 nM T46360 C34VIY 77042 IC50 > 5000 nM T46360 C0QAT3 88747 Ki > 10000 nM T46360 CB3U0P 90748 Ki = 0.67 nM T46360 CN26SL 93365 Ki = 0.01 nM T46360 C3JXH7 97478 Ki = 1150 nM T46360 CI8KD2 97627 Ki = 1480 nM T46360 CA3W0P 100826 IC50 > 100000 nM T46360 CY65GC 112416 IC50 > 10000 nM T46360 CW0G3U 119010 IC50 = 56 nM T46360 CM34NA 119265 Ki = 14.34 nM T46360 CT2H5A 121180 IC50 = 362 nM T46360 C21KTQ 121968 Ki = 10 nM T46360 CKR4N3 122065 Ki > 50 nM T46360 C1B4NI 125328 Ki = 2.4 nM T46360 CRJ7G1 126229 Ki = 0.9 nM T46360 C4VK3Y 126260 IC50 = 1.175 nM T46360 CYJ07C 126388 Ki = 0.34 nM T46360 C9BYH2 128032 Ki = 4.3 nM T46360 CE75MR 131253 Ki = 2 nM T46360 CNO1J3 131444 Ki = 17 nM T46360 CU0C6S 131698 Ki = 2.7 nM T46360 CUYI35 132954 IC50 = 3.47 nM T46360 C2KAL0 132995 Ki = 1.7 nM T46360 C85AXM 164487 IC50 = 26 nM T46360 C7QCS6 185717 IC50 = 50 nM T46360 C3SG4X 185834 Ki = 0.04 nM T46360 CFAP45 190868 Ki = 0.05 nM T46360 CNJ78I 192277 IC50 = 3020 nM T46360 CZDX91 192370 Ki = 168 nM T46360 C9Z3NL 192481 Ki = 10.4 nM T46360 CI9E2D 192611 IC50 = 0.29 nM T46360 CA3T7R 192638 IC50 = 228 nM T46360 CD19AW 192639 IC50 = 33 nM T46360 C5KHP9 200601 Ki = 5.81 nM T46360 CU2RH4 202478 Ki = 6 nM T46360 CDM25N 230867 IC50 > 10000 nM T46360 CF16XZ 242976 IC50 = 1370 nM T46360 C9EHT7 252230 IC50 = 15 nM T46360 C39OMI 269722 Ki = 5850 nM T46360 C0PUC2 344343 IC50 = 133 nM T46360 CZEG20 356862 IC50 = 2005 nM T46360 C30GUQ 381254 Ki = 1.64 nM T46360 C0DE9F 381255 Ki = 3.02 nM T46360 C5D4YG 398371 Ki = 720 nM T46360 C5JG2Z 398373 Ki = 2230 nM T46360 C13BVL 398418 Ki = 1100 nM T46360 CW0DY3 398578 Ki = 1.49 nM T46360 CXO6I9 398580 Ki = 1122 nM T46360 C7D0YB 398582 Ki = 77.5 nM T46360 C7QE8N 398586 Ki = 13.8 nM T46360 C01HIV 398588 Ki = 8 nM T46360 C3ZF6U 398839 Ki = 869 nM T46360 CM71EX 401804 Ki = 2220 nM T46360 C9AOD7 401806 Ki = 5460 nM T46360 C95KEG 401808 Ki = 3100 nM T46360 CNAU07 401810 Ki = 276 nM T46360 C3I7AM 401812 Ki = 291 nM T46360 CZLP87 401816 Ki = 579 nM T46360 C7EIT9 401818 Ki = 56 nM T46360 C29XHP 401820 Ki = 26 nM T46360 CH35LT 401822 Ki = 13 nM T46360 CCF24R 401826 Ki = 8.2 nM T46360 C27VBR 401827 Ki = 2.2 nM T46360 CM8JT4 401829 Ki = 1.3 nM T46360 C3AJZ6 401834 Ki = 3.9 nM T46360 CF1IA7 401839 Ki = 1.3 nM T46360 CTMQ39 401843 Ki = 148 nM T46360 CA93IJ 401844 Ki = 4.1 nM T46360 C43UDC 401846 Ki = 2.6 nM T46360 C6KN4X 401850 Ki = 4.1 nM T46360 CM57RI 401854 Ki = 4.8 nM T46360 C8JQ0S 401856 Ki = 2 nM T46360 CD9UV5 401860 Ki = 3.9 nM T46360 C1WEY2 401862 Ki = 1.4 nM T46360 CIX84S 407725 IC50 = 48 nM T46360 C7UEP4 409922 Ki = 7.6 nM T46360 C3HFE4 422923 Ki = 74 nM T46360 CCO6D8 428911 IC50 = 340 nM T46360 C4Y0ME 442108 Ki = 8554 nM T46360 C90GUY 473059 Ki = 72 nM T46360 C06MHS 473073 Ki = 47 nM T46360 CVZ3N0 547467 Ki = 2.3 nM T46360 CB8J6E 558800 Ki = 1.47 nM T46360 CKI0U2 558843 Ki = 4.22 nM T46360 C6AVL5 566741 Ki = 3.69 nM T46360 C4GF6U 573546 Ki = 2.67 nM T46360 CRMK45 573661 Ki = 3.56 nM T46360 CTW61R 574780 Ki = 6.3 nM T46360 CX5W2H 587944 Ki = 0.31 nM T46360 C5P9MF 594236 Ki = 0.39 nM T46360 C1Q3GW 604376 Ki = 0.52 nM T46360 C82CBK 620985 IC50 = 83 nM T46360 CJL68V 648525 IC50 = 1480 nM T46360 C35WDY 659840 Ki = 26 nM T46360 CQD2N8 728567 IC50 = 3500 nM T46360 C74ZXL 743379 Ki = 6.7 nM T46360 CU1R0C 762654 Ki = 11360 nM T46360 C80NWF 762919 Ki = 0.47 nM T46360 CQJW96 763622 Ki = 0.39 nM T46360 CRBO37 764022 Ki = 0.58 nM T46360 CUE5T3 764613 Ki = 1.4 nM T46360 CTF1D3 764825 Ki = 5.3 nM T46360 CM6Z0W 765219 Ki = 0.46 nM T46360 C8HU1D 782728 Ki = 706 nM T46360 C5S3MB 785789 Ki = 3.8 nM T46360 CUF0O4 796534 IC50 = 109 nM T46360 CS4XQ9 1081502 Ki > 100 nM T46360 CK04FA 1245023 Ki = 6.46 nM T46360 CK0JI9 1548955 Ki = 5 nM T46360 CUF6Z2 2225138 Ki = 26.9 nM T46360 CT7GF8 2427316 Ki = 0.2089 nM T46360 CHA7K3 2712605 Ki = 3.93 nM T46360 CLU95O 2729533 Ki = 30.8 nM T46360 C8VTI5 2817997 Ki = 3.9 nM T46360 CF96BK 2845469 Ki = 10.5 nM T46360 CZ7C0Q 2845594 Ki = 7.5 nM T46360 C9FHM1 3035672 Ki = 0.8 nM T46360 CM3GY5 3036027 Ki = 1.3 nM T46360 C2TAD3 3036289 Ki = 696 nM T46360 C4TB0I 3036864 IC50 = 389.05 nM T46360 CZPH80 3037711 Ki = 82.9 nM T46360 CLB7W5 3037886 Ki = 2100 nM T46360 CE4KC8 3038603 Ki = 800 nM T46360 C54FEG 3039881 Ki = 550 nM T46360 C7MQC0 3041078 Ki = 482 nM T46360 C6RJ5X 3043720 Ki = 22 nM T46360 C6Z4QI 3050372 Ki = 77.1 nM T46360 CI5W4L 3064081 IC50 > 10000 nM T46360 C5NA6S 3069135 Ki = 41.5 nM T46360 CJ7K3Y 3081049 Ki = 3720 nM T46360 CNL68D 3083456 IC50 = 4 nM T46360 C2SE0V 3083457 IC50 = 0.5 nM T46360 CS5F1I 3083481 Ki = 4.4 nM T46360 C6AX8Y 3126148 Ki > 100 nM T46360 C0WFU5 3296345 Ki = 66.4 nM T46360 CJ4Y7Q 3299322 Ki = 2.9 nM T46360 C6G4UP 3315413 IC50 = 140 nM T46360 CJ6D8N 3342390 Ki < 1000 nM T46360 C7V3QI 3562491 Ki = 22.66 nM T46360 CE49MQ 3869448 Ki = 1.46 nM T46360 CGUE70 4033090 Ki = 6.65 nM T46360 CW9SC1 4058484 IC50 > 10000 nM T46360 CWX41S 4598397 Ki = 12 nM T46360 CRM98I 4687238 IC50 = 0.7244 nM T46360 CO84FU 4827344 Ki = 9.66 nM T46360 C47FSG 4879851 Ki = 10.1 nM T46360 CO30PB 4992580 Ki = 19.2 nM T46360 CZF7B5 5026275 Ki = 0.17 nM T46360 C2M4DQ 5221975 Ki = 3.9 nM T46360 C4J7FP 5236783 Ki = 4.89 nM T46360 CK8D2C 5370189 Ki = 0.86 nM T46360 CR4G2N 5461916 Ki = 0.67 nM T46360 C95ADL 5468874 Ki = 7436 nM T46360 CVCA38 5468876 Ki = 27.3 nM T46360 C2DNO0 5471948 Ki = 2.4 nM T46360 C97VGU 5474589 Ki = 3 nM T46360 C0J2GT 5478726 Ki = 1.3 nM T46360 C6ZL2O 5974189 IC50 = 51 nM T46360 CFGZ19 6273133 Ki = 3.2 nM T46360 CB3M8S 6331636 Ki = 455 nM T46360 C9J6HG 6430604 Ki = 275 nM T46360 CFO08L 6437849 Ki = 680 nM T46360 C2UV7A 6439331 Ki = 3 nM T46360 CIPW27 6465840 Ki = 30.1 nM T46360 CGM63Y 6540428 IC50 = 912.01 nM T46360 CED0X6 6604724 Ki = 594 nM T46360 C5WH0F 6604868 IC50 = 28 nM T46360 C6R4WZ 6712729 Ki = 11.2 nM T46360 CCU3H5 6712751 IC50 = 278 nM T46360 C9G5RB 6712752 IC50 = 128 nM T46360 C1M9QS 6713949 Ki = 81 nM T46360 C0S1MT 6918656 Ki = 4.3 nM T46360 C1ORF3 6995232 Ki = 1258.93 nM T46360 C4Z0DT 9049339 Ki = 2.1 nM T46360 CCN7X5 9208936 Ki = 3.97 nM T46360 C9UB2N 9795762 Ki = 10 nM T46360 C4V0PN 9796317 Ki = 5.4 nM T46360 C24EXG 9796923 Ki = 0.51 nM T46360 CK3DI8 9797419 Ki = 6.59 nM T46360 CNXS47 9797436 Ki = 1.39 nM T46360 CDT7Q4 9797984 IC50 = 10700 nM T46360 CD8H3W 9799239 Ki = 0.5 nM T46360 CPB9S2 9800653 IC50 = 7551 nM T46360 CXI46Z 9802946 Ki = 13.82 nM T46360 C32AXD 9803895 Ki = 2.25 nM T46360 C7R0UJ 9804703 Ki = 3.21 nM T46360 CN2XR0 9817442 IC50 = 54 nM T46360 C0XJ8E 9817503 IC50 = 5.888 nM T46360 C2FVL8 9818804 IC50 = 16 nM T46360 CWJB39 9819510 Ki = 6.3 nM T46360 CJ96KD 9820591 Ki = 4.4 nM T46360 CH60LU 9823429 IC50 = 1.8 nM T46360 C82CXQ 9835629 IC50 = 1860 nM T46360 C73NUA 9835807 IC50 = 362 nM T46360 C5EDO7 9839491 Ki = 1 nM T46360 C9PC6E 9839973 IC50 = 2190 nM T46360 CHSR07 9840044 Ki = 56 nM T46360 C26QDV 9840310 Ki = 8.22 nM T46360 CXYJ93 9841596 Ki = 1 nM T46360 C89FSJ 9841846 Ki = 1.15 nM T46360 C3FK5G 9847317 Ki = 81 nM T46360 C6CXW8 9858146 IC50 = 1210 nM T46360 C17IQN 9861694 Ki = 4.3 nM T46360 CGC5E7 9862757 IC50 = 1000 nM T46360 CTF7N5 9863340 Ki = 2 nM T46360 C0BQA3 9864023 Ki = 14 nM T46360 CBW2I4 9864749 Ki = 0.67 nM T46360 C5XBP1 9868470 Ki = 4.2 nM T46360 C2V9FQ 9882367 Ki = 1.11 nM T46360 CAI67X 9882743 Ki = 654 nM T46360 CX8M6A 9883221 Ki = 2 nM T46360 C40DMV 9883360 Ki = 0.26 nM T46360 CX9P2S 9883361 Ki = 1.48 nM T46360 CI2R9W 9883362 Ki = 0.83 nM T46360 CL5V6S 9883820 Ki = 10.16 nM T46360 C3DB5H 9884781 Ki = 1.6 nM T46360 CTAC24 9885114 Ki = 232 nM T46360 CP1GD3 9887523 Ki = 1.21 nM T46360 C2S8KJ 9889112 Ki = 6.75 nM T46360 CA7F6X 9889113 Ki = 9.03 nM T46360 CHB63J 9889709 Ki = 4.8 nM T46360 CTY4K6 9890959 IC50 = 43 nM T46360 CL0Z7Q 9902485 IC50 = 6130 nM T46360 CNO38Q 9905222 Ki = 7 nM T46360 C4UP3E 9905985 Ki = 0.49 nM T46360 CH7K4W 9906138 Ki = 5.51 nM T46360 CAEG95 9906139 Ki = 3.15 nM T46360 CYWQ50 9906447 Ki > 10000 nM T46360 C9XIG6 9919363 IC50 = 13 nM T46360 C7PC1V 9921810 IC50 = 82 nM T46360 C0UH2P 9923341 IC50 = 4800 nM T46360 CY3FW6 9924349 Ki = 3.3 nM T46360 CV28TC 9925741 Ki = 0.25 nM T46360 C85CAL 9926814 Ki = 0.98 nM T46360 CAY53L 9927364 Ki = 3.56 nM T46360 CS29LN 9927617 Ki = 1300 nM T46360 CBSW20 9930604 Ki = 288.4 nM T46360 C1UA3Y 9936242 Ki = 1.78 nM T46360 CSH40U 9936494 IC50 = 183 nM T46360 CN59VH 9943903 IC50 = 2.754 nM T46360 C78DMI 9951886 Ki = 1.3 nM T46360 CZ0AT6 9954083 Ki = 1 nM T46360 CIT01A 9956313 IC50 > 100 nM T46360 CKMW59 9957260 Ki = 110 nM T46360 CNB8Q5 9966844 IC50 = 6260 nM T46360 CDR7Y4 9970628 IC50 = 2900 nM T46360 C9OM2Z 9973696 Ki = 1.75 nM T46360 CPY61E 9973880 Ki = 40.7 nM T46360 CUHA14 9974013 IC50 = 965 nM T46360 CFSR80 9975973 IC50 = 52 nM T46360 C5VNI2 9981159 Ki = 66.2 nM T46360 CIP7Q9 9992101 Ki = 0.07 nM T46360 CFE9H1 9994390 IC50 = 2700 nM T46360 CE3HF7 9995041 IC50 = 240 nM T46360 C4CYX9 9996818 IC50 = 2290 nM T46360 C5AO4D 9998085 Ki = 4 nM T46360 C6WY0U 9999116 Ki = 21.6 nM T46360 C9T0UJ 9999184 IC50 = 320 nM T46360 CXU2V1 10001045 Ki = 128 nM T46360 C6QPD3 10001759 Ki = 76.9 nM T46360 CIZ3D8 10001888 Ki = 110 nM T46360 CX36LV 10002293 Ki = 0.65 nM T46360 CQ5NZ7 10016031 IC50 = 351 nM T46360 C97KHW 10017418 Ki = 2.7 nM T46360 CQH60R 10017724 Ki = 16.05 nM T46360 CG0IW7 10017936 Ki = 0.6 nM T46360 C1XK9Y 10019102 Ki = 1.29 nM T46360 C9LC6Z 10020651 IC50 = 140 nM T46360 C94EDH 10021099 Ki = 2 nM T46360 CQ9M7E 10021279 Ki = 2.5 nM T46360 C7HU5C 10021562 IC50 = 54.4 nM T46360 CS83XQ 10022628 Ki = 46 nM T46360 CFB0D2 10023021 Ki = 3.11 nM T46360 C3RH0Z 10023073 Ki = 0.87 nM T46360 CU93MX 10023529 Ki = 0.46 nM T46360 CL5IW1 10024634 Ki = 1.34 nM T46360 CB5T9V 10025360 IC50 = 1034 nM T46360 CSI9J6 10025403 Ki = 6.9 nM T46360 CI92JG 10025852 Ki = 16.53 nM T46360 CF6O3E 10027435 Ki = 2 nM T46360 CXZ3Q6 10037913 IC50 = 6280 nM T46360 C3S0HG 10037914 IC50 = 247 nM T46360 CFAO01 10038412 IC50 = 7180 nM T46360 C3Z4OD 10040286 Ki = 12 nM T46360 CZ2IY1 10041139 IC50 = 92 nM T46360 C5KGS0 10041278 Ki = 310 nM T46360 CY6HM5 10041770 Ki = 12.83 nM T46360 CM3L5T 10041887 Ki = 4 nM T46360 C3RPO9 10042466 Ki = 8 nM T46360 CCK0P4 10042708 Ki = 2.89 nM T46360 CIBU84 10043468 Ki = 1.9 nM T46360 CJ3V7G 10045023 Ki = 26 nM T46360 CZGN76 10048702 Ki = 335 nM T46360 C9B8JP 10049124 Ki = 16 nM T46360 C4T1PW 10061124 Ki = 21.66 nM T46360 CE4GX6 10064346 IC50 = 2740 nM T46360 CP0K9A 10064484 Ki = 1.54 nM T46360 C6V0IR 10064992 Ki = 4.34 nM T46360 C8FLO9 10065022 Ki = 440 nM T46360 CDX32I 10065362 Ki = 1.53 nM T46360 CP1S7J 10066063 Ki = 26.6 nM T46360 COZU58 10066419 Ki = 7 nM T46360 C0ISR6 10067170 Ki = 15 nM T46360 CU18XB 10069224 Ki = 25 nM T46360 CO69FB 10069973 Ki = 4295 nM T46360 C24TYX 10070045 IC50 = 92.8 nM T46360 CG5B2A 10070289 IC50 = 138 nM T46360 CQV2B9 10074800 Ki = 1.44 nM T46360 CI3D4F 10085466 Ki = 1.48 nM T46360 CI3R6W 10085970 Ki = 8.9 nM T46360 CROI43 10086447 Ki = 167 nM T46360 C9ECP3 10086666 Ki = 2.17 nM T46360 C9DX0V 10087782 Ki = 12 nM T46360 CVG5X1 10087999 Ki = 54 nM T46360 CIMQ96 10090127 Ki = 13 nM T46360 CKO26X 10090269 IC50 = 125 nM T46360 CU70GB 10090882 IC50 = 2100 nM T46360 CS3W1Z 10091077 Ki = 62.8 nM T46360 C7O8VH 10092041 IC50 = 64.1 nM T46360 CV48RC 10094571 Ki = 0.27 nM T46360 C0B8NJ 10094793 IC50 = 62 nM T46360 C1US0Q 10106826 Ki = 1.35 nM T46360 CRM6E0 10107042 Ki = 1.3 nM T46360 CM09JQ 10107360 Ki = 62.06 nM T46360 C6A5MJ 10107472 Ki = 243 nM T46360 CN4PY7 10108342 IC50 = 29 nM T46360 CQCN30 10108347 Ki = 26.7 nM T46360 CYKX67 10149140 Ki = 117 nM T46360 CTQ2A6 10176973 IC50 = 10.96 nM T46360 CZKG96 10200496 Ki = 3.4 nM T46360 C8R2AC 10243335 IC50 = 43 nM T46360 C51YTO 10243428 Ki = 7280 nM T46360 C31ZJX 10243991 IC50 = 1070 nM T46360 CKLA98 10246015 Ki = 410 nM T46360 C0NT8I 10248163 IC50 = 99.1 nM T46360 C0E5SL 10248164 IC50 = 246 nM T46360 C0UQ6P 10250792 IC50 = 53.5 nM T46360 CY9KM2 10250837 Ki = 1.02 nM T46360 CR4C1F 10253032 Ki = 5160 nM T46360 C6JH3D 10254219 Ki = 227 nM T46360 C4TK2U 10263215 Ki = 1042 nM T46360 CD5GU8 10263742 Ki = 1130 nM T46360 CWC2I4 10264753 Ki = 2.17 nM T46360 C48VLE 10264983 Ki = 6.6 nM T46360 CQJZ52 10264992 Ki = 1.18 nM T46360 CI29SE 10265752 Ki = 0.5 nM T46360 C1OER8 10266406 Ki = 21.3 nM T46360 C2F4ON 10266413 Ki = 0.69 nM T46360 CWF4D9 10267592 Ki = 710 nM T46360 CCP61G 10267880 IC50 = 7250 nM T46360 CW6UR5 10271046 IC50 = 234 nM T46360 C36PLT 10313891 Ki = 4 nM T46360 CP3Q4V 10314247 Ki = 1.45 nM T46360 CU3AC0 10314788 Ki = 10 nM T46360 CZM6T1 10316192 Ki = 11 nM T46360 CQZV80 10316321 Ki = 2.5 nM T46360 C7Q9KA 10319121 Ki = 0.51 nM T46360 C59KRL 10319931 Ki = 0.61 nM T46360 CNW60B 10331008 Ki = 83 nM T46360 CZ7AR2 10331473 Ki = 0.48 nM T46360 C34EYX 10333740 Ki = 0.96 nM T46360 C4K9SA 10334147 Ki = 21 nM T46360 CMX6Y0 10334410 Ki = 13 nM T46360 CARB42 10335164 Ki = 0.34 nM T46360 CT41RK 10336644 Ki = 9.6 nM T46360 C70MLB 10337045 Ki = 3 nM T46360 C5OT2E 10337119 Ki = 512.86 nM T46360 C60KJG 10337232 Ki = 265 nM T46360 CZI96H 10338172 Ki = 0.72 nM T46360 C3YCB5 10339444 Ki = 20.5 nM T46360 C2OCU0 10339767 Ki = 3 nM T46360 C9LKM0 10340180 IC50 = 7930 nM T46360 CO7C5M 10341072 Ki = 1.3 nM T46360 CF2U7Y 10342248 Ki = 2.78 nM T46360 C8KX0R 10342773 IC50 = 87.5 nM T46360 CF6NS0 10342845 Ki = 1.21 nM T46360 CS6P0J 10344430 Ki = 372 nM T46360 C52ZML 10354750 Ki = 6 nM T46360 CUK08H 10356159 Ki = 4.3 nM T46360 CZ9MG4 10356384 Ki > 100 nM T46360 CLG82T 10356463 Ki = 153 nM T46360 CN8PA7 10357986 Ki = 1.14 nM T46360 C6ZN0S 10358634 IC50 = 2640 nM T46360 CUD17B 10358719 Ki = 0.09 nM T46360 CG9WL5 10361439 IC50 = 198 nM T46360 C50OXW 10361564 Ki = 5 nM T46360 CW65RM 10365559 Ki = 27.22 nM T46360 CV2IT8 10365874 Ki = 1.3 nM T46360 C4I9US 10367771 Ki = 386.37 nM T46360 CM64TP 10368819 Ki = 22.8 nM T46360 CVY37K 10369311 Ki = 6 nM T46360 CWX81D 10369315 Ki = 0.88 nM T46360 CAYV90 10376919 Ki = 7.4 nM T46360 C9AJ7X 10378304 IC50 = 8 nM T46360 CO8NE3 10378306 IC50 = 1410 nM T46360 C2H1OB 10380647 Ki = 0.5 nM T46360 C7G9TF 10382446 Ki = 9 nM T46360 CYZN57 10383371 Ki = 2.19 nM T46360 CON6G8 10384067 IC50 = 55 nM T46360 CCZ74R 10384372 Ki = 9 nM T46360 CLY48W 10385977 IC50 = 59.9 nM T46360 C76DIU 10389641 IC50 = 707 nM T46360 C4DZ0M 10392655 Ki = 809 nM T46360 C34TLK 10402464 Ki = 1.34 nM T46360 C5SGY8 10404406 Ki = 13.4 nM T46360 C58RMD 10405079 Ki = 2.37 nM T46360 CHK46F 10405640 Ki = 101.7 nM T46360 CO34LY 10405821 IC50 = 8480 nM T46360 CDI85V 10406366 IC50 = 173 nM T46360 C5J6ZM 10407855 IC50 = 40 nM T46360 CKWY76 10408160 Ki = 0.5 nM T46360 CB67IL 10410177 Ki = 1.51 nM T46360 CZR8Q9 10422239 Ki = 5.4 nM T46360 CX1FR6 10423970 Ki = 26 nM T46360 C3JZ5Y 10426298 Ki = 16.76 nM T46360 CEKH47 10426373 Ki = 27 nM T46360 CLE64B 10426722 IC50 = 343 nM T46360 C2ZOF1 10428881 Ki = 46.98 nM T46360 CG0QM1 10429420 Ki = 24 nM T46360 C1A8XG 10430305 Ki = 19 nM T46360 CA1FD2 10430685 Ki = 61 nM T46360 C8Q4BP 10432985 Ki = 929.72 nM T46360 CN62ZX 10436105 Ki = 283 nM T46360 C1ZB7H 10446096 IC50 = 75 nM T46360 CO3EC1 10446949 IC50 = 13000 nM T46360 C36NJX 10447715 IC50 = 91 nM T46360 CBNM05 10447949 IC50 = 60 nM T46360 CS6E1O 10448420 Ki = 580 nM T46360 CYW8U4 10448771 Ki = 2.08 nM T46360 CMFL03 10449500 Ki = 9.4 nM T46360 CF25ZL 10449555 Ki = 2.66 nM T46360 CI0N2R 10449738 Ki = 11 nM T46360 CCP2O7 10450158 Ki = 3.6 nM T46360 C2G0AH 10450758 Ki = 35 nM T46360 C78IQN 10451373 Ki = 1066 nM T46360 CLY07Z 10453320 IC50 = 151 nM T46360 CACD15 10453690 IC50 = 11000 nM T46360 CAM7K8 10458892 Ki = 12900 nM T46360 CM48KH 10466885 Ki = 4450 nM T46360 C10HGT 10467460 Ki = 11.4 nM T46360 C6I2JZ 10467461 Ki = 4.8 nM T46360 C1B0JC 10470687 Ki = 4.3 nM T46360 CLE8W0 10470688 Ki = 2.9 nM T46360 C3BSH7 10473287 Ki = 1.2 nM T46360 C7GEB0 10474042 IC50 = 67.5 nM T46360 CTB5N8 10474751 Ki = 3.95 nM T46360 C8KE2J 10475196 Ki = 37 nM T46360 CUE5J0 10475634 IC50 = 52.2 nM T46360 C9S0EG 10491108 IC50 = 42.8 nM T46360 CLQU72 10493098 IC50 = 20.6 nM T46360 CIK95Q 10496036 IC50 > 1000 nM T46360 COES83 10496045 IC50 = 28.5 nM T46360 CU3GS8 10496297 IC50 = 110 nM T46360 C23KXT 10497826 Ki = 1.54 nM T46360 CU49FK 10498073 Ki = 29.6 nM T46360 CDMT59 10498740 IC50 = 65 nM T46360 COE3F4 10499273 Ki = 43.4 nM T46360 CI3TV1 10501583 Ki = 1.32 nM T46360 C4ZK6D 10502049 IC50 = 1050 nM T46360 C69BVP 10503221 IC50 = 150 nM T46360 CG72YU 10503374 IC50 = 8.6 nM T46360 C6K4WF 10504449 IC50 > 1000 nM T46360 C5HOS1 10517426 IC50 = 71.8 nM T46360 C30UGV 10517496 Ki = 19.8 nM T46360 CC94RX 10518276 IC50 = 164 nM T46360 C25ZVH 10521200 Ki = 20 nM T46360 C5NJ9X 10522573 Ki = 0.63 nM T46360 CFE07M 10522765 IC50 = 10 nM T46360 C9SGF2 10522997 Ki = 7.9 nM T46360 C3ZE8F 10524644 Ki = 1500 nM T46360 CXLS06 10525997 Ki = 4 nM T46360 C8Q0AM 10539358 Ki = 181 nM T46360 C94PRD 10540231 IC50 = 15.9 nM T46360 C9QX7K 10540232 IC50 = 20 nM T46360 C7XG2K 10541325 IC50 = 43.5 nM T46360 CK1IJ0 10542038 Ki = 62.3 nM T46360 C9NU4M 10542799 IC50 = 36.5 nM T46360 CJ7CY6 10545203 IC50 = 8 nM T46360 CA4P0N 10546938 Ki = 7.6 nM T46360 CKD9N5 10546961 Ki = 18.4 nM T46360 C5EJ9T 10550623 Ki = 31 nM T46360 CQD6C8 10551026 Ki = 5.9 nM T46360 CK27CJ 10551210 IC50 = 180 nM T46360 CEP7J1 10551313 Ki = 57 nM T46360 CZT94B 10564492 Ki = 7.7 nM T46360 C2PIU7 10564493 Ki = 6.4 nM T46360 CACP09 10566716 IC50 = 11.8 nM T46360 CJRB30 10567286 Ki = 127 nM T46360 CUR2O0 10568910 Ki = 61.66 nM T46360 C6OJL3 10569632 Ki = 6.457 nM T46360 CE2AQ9 10570139 Ki = 5.3 nM T46360 CO8SK3 10571211 Ki = 32.1 nM T46360 CD80FJ 10571528 Ki = 86 nM T46360 C10GOH 10575209 IC50 = 78 nM T46360 C2FAG0 10582642 Ki = 1.2 nM T46360 C1JH4Y 10582670 Ki = 1.9 nM T46360 CT78EI 10587586 Ki = 30.3 nM T46360 COR05F 10587917 IC50 = 18.5 nM T46360 CLD91R 10589924 Ki = 5.012 nM T46360 C9YSV1 10592242 Ki = 3.43 nM T46360 CW1L0N 10593974 IC50 = 330 nM T46360 C2WKD7 10594382 Ki = 63.9 nM T46360 C30YWC 10595615 Ki = 0.18 nM T46360 CONJ90 10596136 Ki = 16.6 nM T46360 CTJ5P1 10598454 IC50 = 381 nM T46360 CQ2M1Y 10599447 Ki = 18 nM T46360 CX1TS7 10599695 IC50 = 79 nM T46360 C9L0WQ 10599798 IC50 = 230 nM T46360 C4N7QJ 10599997 Ki = 1.1 nM T46360 CBAY37 10614630 Ki = 628 nM T46360 CXA13I 10615294 IC50 = 156 nM T46360 CAES37 10615793 IC50 = 97 nM T46360 CIQX09 10616126 Ki = 2.45 nM T46360 CS81FH 10616210 IC50 = 160 nM T46360 C42HFS 10616657 Ki = 115 nM T46360 CJ8T3N 10616816 IC50 > 1000 nM T46360 CG2RS0 10616993 Ki = 10.5 nM T46360 C8EH7Y 10617417 Ki = 7.63 nM T46360 CAT71Z 10618129 Ki = 145 nM T46360 CR5PI7 10618199 IC50 = 170 nM T46360 CZW69I 10618791 Ki = 42.2 nM T46360 CGJ0K6 10618918 Ki = 110.4 nM T46360 CSH12T 10619110 Ki = 29 nM T46360 C05AEY 10619619 Ki = 469 nM T46360 C8EX2V 10619631 IC50 = 130 nM T46360 CX7Q1J 10621853 IC50 = 34 nM T46360 CRS76W 10622914 Ki = 3.2 nM T46360 C7DQP5 10632134 Ki = 14280 nM T46360 C0UM2L 10634649 IC50 = 10.8 nM T46360 CCH7P1 10635235 Ki = 15.7 nM T46360 CAYM59 10635279 Ki = 63 nM T46360 CUE1G6 10637326 Ki = 736 nM T46360 CXO8K0 10638488 IC50 = 69.9 nM T46360 CFS6L3 10639616 Ki = 338.84 nM T46360 CGJ1U0 10640585 IC50 = 39.3 nM T46360 CE4UO3 10641401 Ki = 137.7 nM T46360 CI7T6M 10641797 Ki = 2.6 nM T46360 CO6TF0 10642179 Ki = 23.8 nM T46360 C7AZL4 10642861 IC50 = 420 nM T46360 CS46DA 10644162 Ki = 28 nM T46360 C3AGQ5 10645614 Ki = 0.7 nM T46360 CIN2U8 10646068 IC50 = 170 nM T46360 C4X8HV 10650002 IC50 = 4001 nM T46360 C2PGB1 10660038 Ki = 177 nM T46360 CAI09V 10661409 Ki = 0.6166 nM T46360 CW1H2S 10662563 IC50 = 14.4 nM T46360 C9PR7I 10662728 Ki = 365 nM T46360 C4AU9T 10663237 Ki = 15.2 nM T46360 CY9AE7 10664642 Ki = 5.9 nM T46360 CNX7J5 10665130 Ki = 3.87 nM T46360 CM1V7L 10665131 Ki = 3.17 nM T46360 CFX47R 10666733 Ki = 352 nM T46360 C0RBZ3 10666808 IC50 = 12 nM T46360 CXLA63 10668517 IC50 = 9 nM T46360 C1GPV6 10669784 IC50 = 1.5 nM T46360 CYF30E 10683536 IC50 > 1000 nM T46360 C8WEA9 10684798 Ki > 877 nM T46360 CVJ8N5 10686220 IC50 = 13.3 nM T46360 CCI6W0 10686221 IC50 = 31.8 nM T46360 C6YEV8 10687454 IC50 = 67 nM T46360 CZ27AV 10687985 IC50 = 40 nM T46360 C3SA7L 10689336 Ki = 7.32 nM T46360 CNK7Q5 10689502 Ki = 27.1 nM T46360 CIO4J5 10691389 IC50 = 5.7 nM T46360 CG01CM 10691769 Ki = 0.32 nM T46360 CBUK71 10695744 IC50 > 1000 nM T46360 CI52BL 10696254 Ki = 16.7 nM T46360 CCWU31 10710332 IC50 = 34 nM T46360 C9A1WC 10710941 IC50 = 39 nM T46360 CREK17 10711065 Ki = 159 nM T46360 CK2Y9B 10711119 Ki = 18.8 nM T46360 C6PJ4G 10711455 IC50 = 241 nM T46360 C4RVY0 10712370 Ki = 1.4 nM T46360 CJI3R5 10712473 Ki = 4.21 nM T46360 CN8S0W 10713214 IC50 = 4.5 nM T46360 C4R9DJ 10713754 Ki = 5.8 nM T46360 C52DUN 10713756 Ki = 1.91 nM T46360 C1VT7F 10714699 Ki = 7 nM T46360 CQ7L4I 10715370 Ki = 6520 nM T46360 C4QS9B 10716035 Ki = 457.09 nM T46360 CL8E5M 10717134 Ki = 21.4 nM T46360 CX05VT 10718443 Ki = 3.11 nM T46360 CYL27S 10718492 Ki = 230 nM T46360 C6Q3JA 10719188 Ki = 400 nM T46360 CG4S2Q 10719189 Ki = 6.2 nM T46360 CZ0A1O 10732853 IC50 = 231 nM T46360 CC84XI 10733148 Ki = 72 nM T46360 C9PES2 10733647 Ki = 70.79 nM T46360 CHO52Y 10733648 Ki = 234.42 nM T46360 C3Q4UE 10735303 IC50 = 125 nM T46360 CPZ24W 10735925 Ki > 1000 nM T46360 C8ONT1 10736122 Ki = 3.08 nM T46360 C1QJ2F 10738317 Ki = 139 nM T46360 C8ZH2S 10738339 Ki = 7.28 nM T46360 CA0Y3H 10739649 Ki = 80 nM T46360 C7QLT2 10741325 Ki = 1.2 nM T46360 C6XW5K 10741970 Ki = 1.7 nM T46360 CQ3F5D 10742360 IC50 = 41 nM T46360 C4L9AI 10742465 IC50 = 38 nM T46360 C08PYV 10754756 IC50 = 27 nM T46360 CL15XF 10757227 Ki = 5.754 nM T46360 C62VKE 10758083 Ki = 0.8 nM T46360 CWXZ23 10759399 Ki = 152 nM T46360 C3IQ9W 10761018 Ki = 7.762 nM T46360 C2COG9 10761980 Ki = 6.761 nM T46360 CPV9U1 10762065 Ki = 9.84 nM T46360 CQ1X0J 10762119 Ki = 5.22 nM T46360 C19OPJ 10763386 Ki = 14.2 nM T46360 C25ECH 10764130 IC50 = 29 nM T46360 CV54GW 10766338 Ki = 59 nM T46360 C7BZV3 10766454 IC50 = 30 nM T46360 CYSB34 10779682 IC50 = 45.7 nM T46360 C3RZF4 10779812 Ki = 202 nM T46360 C6JQ7A 10780443 IC50 > 10000 nM T46360 CN6CQ0 10780604 Ki = 286 nM T46360 CO9GR7 10782120 IC50 = 0.5 nM T46360 CA8IP1 10782132 Ki = 89.13 nM T46360 CJ62FW 10782325 Ki = 25 nM T46360 CN5U4I 10783531 Ki = 41.6 nM T46360 CZ5AK0 10784078 Ki = 5.6 nM T46360 CTU4Z6 10784820 Ki = 175 nM T46360 C57DMC 10787011 IC50 = 9.5 nM T46360 C2NG9Q 10789481 Ki = 1.1 nM T46360 CVT79G 10789674 IC50 = 59 nM T46360 CWJ40X 10789833 Ki = 56 nM T46360 C61YUS 10789834 Ki = 5.6 nM T46360 CN3RH8 10790095 Ki = 12.7 nM T46360 CM5S6D 10802506 Ki = 17.3 nM T46360 CAK53D 10805765 IC50 = 64 nM T46360 CT91OQ 10805927 Ki = 286.5 nM T46360 C0ACQ9 10807028 Ki = 43.8 nM T46360 C6IYD4 10807270 Ki = 20.1 nM T46360 C3VRX8 10807460 Ki = 758.58 nM T46360 CX6U3K 10807863 Ki = 1.8 nM T46360 C8O3ZD 10809006 Ki = 3.1 nM T46360 C1CUE8 10809630 IC50 = 110 nM T46360 C85KYQ 10811587 IC50 = 13 nM T46360 C0J7BR 10811875 Ki = 48 nM T46360 C2TPA5 10814571 Ki = 124.7 nM T46360 C3W7CM 10827238 Ki = 270 nM T46360 C3UHC7 10828366 Ki = 571 nM T46360 CES36I 10829775 Ki = 470 nM T46360 CGR8P0 10829840 Ki = 110 nM T46360 CK92FA 10831286 Ki = 1.2 nM T46360 CD8JF2 10831724 IC50 = 8.5 nM T46360 C6WD3U 10833752 Ki = 4.97 nM T46360 CCFI42 10834075 Ki = 2.89 nM T46360 C6HC0N 10834172 Ki = 9.55 nM T46360 C76JVF 10835756 Ki = 3.6 nM T46360 CRF51E 10835977 Ki = 0.14 nM T46360 CN2P9X 10836067 Ki = 41.8 nM T46360 CV4U5D 10836428 Ki = 5.8 nM T46360 CIBE62 10841374 IC50 = 3640 nM T46360 CAR05H 10849098 Ki = 23.8 nM T46360 CM7E2C 10850173 Ki = 19.6 nM T46360 CS8DX0 10851124 Ki = 1850 nM T46360 CW0P3J 10852782 Ki = 7.4 nM T46360 CJ9IL3 10852997 IC50 = 10.3 nM T46360 C6MC4P 10859662 Ki = 12.6 nM T46360 C62RCN 10862129 Ki = 298.56 nM T46360 C72FGM 10870255 Ki = 248.36 nM T46360 CI20YO 10871797 Ki = 13.3 nM T46360 CT7MS4 10881675 Ki = 1.83 nM T46360 C43WZD 10883323 Ki = 87.05 nM T46360 CRI50E 10885636 IC50 = 702 nM T46360 C5Z0DE 10893870 Ki = 15.1 nM T46360 C4J3YU 10895188 Ki = 51.94 nM T46360 C78FGZ 10902342 Ki = 0.86 nM T46360 C52TBK 10902954 Ki = 298.47 nM T46360 C42LHP 10903339 Ki = 11.7 nM T46360 CX65PW 10907460 IC50 = 482 nM T46360 C4SBO9 10915140 Ki = 2.07 nM T46360 C4L9XY 10924765 Ki = 12 nM T46360 CXO09C 10925078 Ki = 7.2 nM T46360 C8HG0I 10926436 Ki = 61.77 nM T46360 C1T9ZG 10936043 Ki = 2.21 nM T46360 CJA61X 10936501 Ki = 15.9 nM T46360 CA8NR0 10936584 Ki = 55.1 nM T46360 CN4TU6 10937393 Ki = 170 nM T46360 C7ACH1 10946809 Ki = 235.5 nM T46360 C9CEG5 10947083 Ki = 2.69 nM T46360 CB2E6K 10948128 Ki = 8.95 nM T46360 CYS1M8 10948383 IC50 = 158 nM T46360 CO04EB 10948807 Ki = 141.36 nM T46360 CP0J7O 10950137 Ki = 346.9 nM T46360 CBQ2J3 10969171 Ki = 1.4 nM T46360 CZ61YN 10969173 Ki = 1.7 nM T46360 CYB4W9 10969339 Ki = 31.25 nM T46360 C9QBS4 10970390 Ki = 4.64 nM T46360 C5LZH9 10980649 Ki = 6.64 nM T46360 CQ7A1S 10981062 Ki = 3.97 nM T46360 CE5K8F 10991643 Ki = 10.9 nM T46360 C7R1CB 11001837 Ki = 7.27 nM T46360 C0UY4P 11003384 Ki = 183 nM T46360 CJT8Y7 11012319 Ki = 269.15 nM T46360 CJ78DG 11013161 Ki = 12.4 nM T46360 C6YWX4 11013162 Ki = 12.7 nM T46360 CE04WV 11016132 Ki = 2.31 nM T46360 C82RNS 11016707 Ki = 3.49 nM T46360 CQ6M1S 11028157 Ki = 751 nM T46360 CGA2C4 11034660 Ki = 43.7 nM T46360 C89XHJ 11034920 Ki = 1390 nM T46360 C8SH3D 11035595 Ki = 19.07 nM T46360 CB7N1P 11035765 IC50 = 328 nM T46360 CXPD18 11045363 Ki = 1.09 nM T46360 C4LE3O 11046757 Ki = 9.33 nM T46360 C23JHR 11047568 IC50 = 2170 nM T46360 CS9FX5 11064325 Ki = 19800 nM T46360 CGI1R9 11091108 Ki = 13.1 nM T46360 CK2WT1 11102433 Ki = 4.29 nM T46360 CU21VJ 11109490 Ki = 2.18 nM T46360 CF3D0J 11109952 Ki = 2.16 nM T46360 C2MR9D 11110106 Ki = 7.16 nM T46360 CF29UZ 11111624 Ki = 125.41 nM T46360 C65WYU 11120436 Ki = 5.66 nM T46360 CY2N6C 11142430 Ki = 149.84 nM T46360 C49ECI 11143217 Ki = 1.87 nM T46360 C1BIZ9 11143323 Ki = 7.24 nM T46360 CU6PV0 11143820 IC50 = 581 nM T46360 C74YMR 11152920 Ki = 5.54 nM T46360 CYS2X0 11154079 Ki = 1.2 nM T46360 CC1AT3 11165837 Ki = 3078 nM T46360 CMA72C 11168272 Ki = 18 nM T46360 C8SL0F 11189143 Ki = 16.2 nM T46360 CU5ND9 11191741 Ki = 1159 nM T46360 CQ9NP6 11198145 Ki = 2 nM T46360 CK34VH 11199981 Ki = 1.54 nM T46360 CAZ9K5 11233111 Ki = 0.61 nM T46360 C27PSA 11234042 Ki = 3.38 nM T46360 C0UMB4 11234470 Ki = 36.4 nM T46360 CM59CS 11235994 Ki = 15.1 nM T46360 C3NF5Z 11237443 Ki = 15.4 nM T46360 CZKE17 11268724 Ki = 0.36 nM T46360 CUSN36 11281378 Ki = 3.07 nM T46360 CZS56H 11292472 Ki = 1.52 nM T46360 CQ0FP3 11292970 Ki = 10000 nM T46360 CGZM12 11302686 Ki = 0.036 nM T46360 CQ29OL 11303155 Ki = 1.45 nM T46360 CQ2Z6J 11304676 Ki = 276.5 nM T46360 CBAU26 11315257 Ki = 21.8 nM T46360 C0LVZ4 11317999 Ki = 189.1 nM T46360 CJT02X 11326158 Ki = 28.7 nM T46360 CTIX74 11338096 Ki = 10400 nM T46360 C3JBI0 11338418 Ki = 0.3 nM T46360 CL7O2I 11349674 Ki = 9.4 nM T46360 CENY72 11360254 Ki > 1000 nM T46360 CY20HV 11372576 Ki = 9.9 nM T46360 CN96RT 11381875 Ki = 0.4 nM T46360 C3V7NH 11405584 Ki = 1.5 nM T46360 C17XGQ 11405620 Ki = 1.57 nM T46360 CGH8L0 11405872 Ki = 2.4 nM T46360 C6WM2A 11406043 Ki = 1.4 nM T46360 CMI90K 11407131 Ki = 0.3 nM T46360 C7CX1Z 11407133 Ki = 0.4 nM T46360 C4HVO6 11416825 Ki = 0.22 nM T46360 CGA4V6 11428574 Ki = 1.57 nM T46360 CGU24X 11428679 Ki = 2.45 nM T46360 C7GB8T 11439301 Ki = 0.31 nM T46360 C2B9FV 11440556 Ki = 36.3 nM T46360 CJW6P0 11451147 Ki = 0.69 nM T46360 C6GXJ4 11451971 Ki = 11.9 nM T46360 CL61VY 11462448 Ki = 5.4 nM T46360 CAL0Z7 11488451 Ki = 2932 nM T46360 CVU67H 11494142 Ki = 17.2 nM T46360 CUTX86 11494380 Ki = 6.9 nM T46360 CQX19K 11501260 Ki = 10.4 nM T46360 C0KBI1 11501613 Ki = 8.2 nM T46360 CN0OV4 11508643 Ki = 5.5 nM T46360 CCQ5N8 11518209 Ki = 26 nM T46360 C5MRO3 11522946 Ki = 5.2 nM T46360 CN35YZ 11531125 Ki = 10.2 nM T46360 CBFZ60 11531451 Ki = 4 nM T46360 C0HL2V 11531518 Ki = 24 nM T46360 CWXL39 11532920 Ki = 16 nM T46360 CB6PI4 11537339 Ki = 10 nM T46360 CVUI98 11544226 Ki > 1000 nM T46360 CU3Z9X 11544597 Ki = 294 nM T46360 C5TZV9 11552718 Ki = 13.3 nM T46360 CY1H3V 11558654 IC50 = 15.5 nM T46360 C26EIT 11567446 Ki = 9.9 nM T46360 COPG87 11573361 Ki = 7 nM T46360 C3UQL8 11573971 Ki = 10.8 nM T46360 CFT29G 11594918 Ki = 9.9 nM T46360 C65ESO 11602582 Ki = 9.9 nM T46360 C9XM1Q 11604103 Ki = 224 nM T46360 C0TAC4 11610271 Ki = 854 nM T46360 C51DOW 11617627 Ki = 17.6 nM T46360 CUCN59 11618199 Ki = 741 nM T46360 C8IE7O 11624298 Ki = 8.2 nM T46360 CPA75G 11625126 Ki = 7.1 nM T46360 CO19EP 11632093 Ki = 11.7 nM T46360 CW42YV 11646372 Ki = 11.1 nM T46360 CES7K4 11652595 IC50 = 11.3 nM T46360 C8B5GK 11652762 Ki = 15.7 nM T46360 C1HDM5 11653679 Ki = 23.44 nM T46360 C8EHT5 11659822 Ki = 47 nM T46360 CFB42T 11667265 Ki = 16.7 nM T46360 CO23PC 11668112 Ki = 172 nM T46360 CN0TZ2 11682186 Ki = 9.4 nM T46360 C3XDB2 11704592 Ki = 44 nM T46360 CF02CY 11704696 Ki > 1000 nM T46360 CWM71X 11718233 Ki = 14.8 nM T46360 C3KU0D 11722772 Ki = 0.49 nM T46360 C6ZGX3 11723852 Ki = 0.97 nM T46360 CME0R3 11725031 Ki = 2 nM T46360 CX1ZF4 11725919 Ki = 29.9 nM T46360 CD9V5B 11733099 Ki = 15.41 nM T46360 CWX41Z 11739209 Ki = 2.16 nM T46360 CDFB43 11743300 Ki = 26700 nM T46360 C1U6PW 11748820 Ki = 29.3 nM T46360 C9GNC5 11758674 Ki = 10100 nM T46360 CBY2Q9 11760579 Ki > 1000 nM T46360 CZ8E3X 11771731 Ki = 125 nM T46360 CDW1T8 11776562 Ki = 28.7 nM T46360 CFSU16 11777643 IC50 = 341 nM T46360 C8DVY0 11777930 Ki = 10 nM T46360 C0P3JO 11782688 Ki = 5.83 nM T46360 CEM4V0 11783308 Ki = 23.88 nM T46360 CJ5Z9H 11784333 Ki = 95.3 nM T46360 CW5L6Q 11791714 Ki = 5.8 nM T46360 C9QI0E 11791902 Ki = 66 nM T46360 CZUE50 11792320 Ki = 54 nM T46360 C6ZQF2 11792374 Ki = 4.56 nM T46360 CWE12Y 11792375 Ki = 18 nM T46360 CZH6S4 11793400 Ki = 121 nM T46360 C3D4PU 11793930 Ki = 8.7 nM T46360 CH6B0Y 11793931 Ki = 3.92 nM T46360 CYR0V7 11794387 IC50 > 1000 nM T46360 C6U2RY 11796923 Ki = 2.5 nM T46360 C9C7HV 11797295 IC50 = 43 nM T46360 C4X8UL 11800052 Ki = 121.8 nM T46360 CHOE91 11808864 Ki = 1.81 nM T46360 CZQ51Y 11810652 Ki = 10.2 nM T46360 CN9M8E 11811722 IC50 = 1250 nM T46360 CT1L3N 11822555 Ki = 7.33 nM T46360 CH91AX 11824300 Ki = 148 nM T46360 CXLW54 11948707 Ki = 180 nM T46360 CT8Q2B 11957591 IC50 = 3.802 nM T46360 CN82RK 11957597 Ki = 118 nM T46360 CKG40P 12084044 Ki = 121 nM T46360 C3ZC4D 12084050 Ki = 69 nM T46360 CCA4D0 12084052 Ki = 96 nM T46360 C6NCO1 12084053 Ki = 28 nM T46360 CE7ZN1 12084054 Ki = 6.2 nM T46360 C6DQ4H 12084055 Ki = 23.4 nM T46360 CZ14EL 12084056 Ki = 375 nM T46360 C5HS8Q 12259685 Ki = 1.7 nM T46360 CSQ2J7 12329382 Ki = 660 nM T46360 C2FOU9 12347284 Ki = 11.7 nM T46360 CA45VN 12351937 Ki = 664 nM T46360 CS5IZ8 12371110 Ki = 6750 nM T46360 CSY9N8 12371111 Ki = 2733 nM T46360 C3Y9UN 12491976 IC50 = 338.84 nM T46360 CQ9F1W 12491977 IC50 = 446.68 nM T46360 C3E7QH 12628908 IC50 = 4100 nM T46360 C2GH7O 12730763 Ki = 20 nM T46360 C4G0MK 12730765 Ki = 29 nM T46360 CH81JK 12730766 Ki = 29 nM T46360 C3H1AN 12874567 Ki = 13.6 nM T46360 CL6G8E 12874569 Ki = 31 nM T46360 CBK95L 12914591 Ki = 48.2 nM T46360 C6LV2S 13011906 Ki = 10.8 nM T46360 C23ELH 13078350 IC50 = 6605 nM T46360 CCG14E 13091356 Ki = 165.96 nM T46360 CYN95Z 13091359 Ki = 81 nM T46360 CYV6B5 13781931 IC50 = 13.8 nM T46360 C2SEG3 13781932 IC50 = 66 nM T46360 CG08MN 13781936 IC50 = 65 nM T46360 C3FCB2 13781939 IC50 = 356 nM T46360 CL7XE8 13998486 Ki = 6 nM T46360 C7VG5C 14040442 IC50 = 1516 nM T46360 CX20PD 14125583 IC50 = 32 nM T46360 CS61DC 14291221 Ki = 418 nM T46360 CJNM56 14292033 IC50 = 220 nM T46360 CC8A3Q 14368937 Ki = 21 nM T46360 CQ9G0L 14368954 Ki = 7 nM T46360 CIE32U 14368960 Ki = 12 nM T46360 CYW76P 14742527 Ki > 1000 nM T46360 C50XLA 14771399 IC50 = 2593 nM T46360 CXM7W9 14771402 IC50 = 418 nM T46360 CA4OM8 14771405 IC50 = 2100 nM T46360 CV87AM 14771416 IC50 = 6058 nM T46360 CNMV48 14771443 IC50 = 77 nM T46360 CDG54I 14771450 Ki = 11 nM T46360 C91VRA 14771452 Ki = 8.66 nM T46360 CHPJ17 14771454 Ki = 1372 nM T46360 CUXT02 14771457 Ki = 456 nM T46360 CA2LP1 14771459 Ki = 7212 nM T46360 C8X7UK 14771468 IC50 = 966 nM T46360 C17WBC 14771473 IC50 = 125 nM T46360 CL7PU3 14771475 IC50 = 37 nM T46360 C6EUR2 14771480 Ki = 89.5 nM T46360 CTAB86 14771482 Ki = 30.5 nM T46360 CRJ0L3 14771666 IC50 = 96 nM T46360 CE0KP4 14771667 IC50 = 59 nM T46360 CM29BA 14771668 IC50 = 36 nM T46360 C5SU1R 14771669 IC50 = 125 nM T46360 CWMO41 14771670 IC50 = 215 nM T46360 CPB79U 14771672 IC50 = 33 nM T46360 C7M1AK 14771673 IC50 = 8110 nM T46360 CTBR56 14771675 IC50 = 203 nM T46360 CQ1ZC3 14771677 IC50 = 16 nM T46360 CX4H7W 14771682 IC50 = 750 nM T46360 CIY37H 14771684 IC50 = 21 nM T46360 CP4LQ5 14771685 IC50 = 37 nM T46360 CR67MN 14771686 IC50 = 42 nM T46360 CEQV06 14771688 IC50 = 440 nM T46360 CH2R4M 14771689 IC50 = 850 nM T46360 CDHN24 14771691 IC50 = 920 nM T46360 C3WK2C 14771692 IC50 = 935 nM T46360 CJ21YE 14771693 IC50 = 1200 nM T46360 CJY5N0 14771694 IC50 = 12 nM T46360 C2NW9K 14771695 IC50 = 6 nM T46360 C47EWB 14771696 IC50 = 8 nM T46360 CF6OB9 14771697 IC50 = 20 nM T46360 CRK3S4 14771698 IC50 = 300 nM T46360 CO4Z3M 14771699 IC50 = 4 nM T46360 C6A4YT 14771702 IC50 = 6 nM T46360 CS9Z3L 14771705 IC50 = 25 nM T46360 C8S0BC 14771707 IC50 = 155 nM T46360 CU94AL 14771709 IC50 = 5.2 nM T46360 C2FO3S 14771711 IC50 = 15 nM T46360 CF2L5J 14771713 IC50 = 16 nM T46360 CL0GD1 14771715 IC50 = 112 nM T46360 C8B9LE 14771717 IC50 = 245 nM T46360 CGJB25 14771719 IC50 = 345 nM T46360 C6JM8H 14771721 IC50 = 370 nM T46360 C0BZJ6 14771723 IC50 = 970 nM T46360 CCW53V 14771725 IC50 = 18 nM T46360 CCMA03 14771728 IC50 = 118 nM T46360 CXGT50 14771729 IC50 = 962 nM T46360 CZSE76 14771731 IC50 = 5100 nM T46360 CCZ3L7 14771734 IC50 = 237 nM T46360 CL7NO6 14771736 IC50 = 238 nM T46360 C64VXZ 14771738 IC50 = 8 nM T46360 CQ92IT 14771742 IC50 = 21.1 nM T46360 C53BMJ 14771744 IC50 > 10000 nM T46360 CDP91Q 14831233 Ki = 9.3 nM T46360 CX7YM2 14831240 Ki = 2.6 nM T46360 CYA34X 14831246 Ki = 97 nM T46360 CXBP45 14831249 Ki = 56 nM T46360 C6CR4J 14895995 IC50 = 10 nM T46360 C42OVT 14941803 Ki = 16.6 nM T46360 C0AY3O 14952694 Ki = 125 nM T46360 CI6MH4 14970526 IC50 = 8 nM T46360 C83VFC 14970527 IC50 = 500 nM T46360 C3MG6W 14970528 IC50 = 100 nM T46360 CKRQ36 14970529 IC50 = 495 nM T46360 C1AYO7 14970530 IC50 = 235 nM T46360 CNF3X6 14970531 IC50 = 400 nM T46360 CA1QS4 14970532 IC50 = 281 nM T46360 C6PO3M 14970533 IC50 = 158 nM T46360 CQ3YR9 14970534 IC50 = 105 nM T46360 CP4G5R 14970535 IC50 = 23 nM T46360 CP6FW7 14970536 IC50 = 25 nM T46360 C6IZC7 14970537 IC50 = 66 nM T46360 CLYJ93 14970538 IC50 = 7 nM T46360 C25QOE 14976641 Ki = 4400 nM T46360 C46ZRG 14977560 IC50 = 140 nM T46360 C3XV5J 14982949 IC50 = 40 nM T46360 CPBC12 14982950 IC50 = 257 nM T46360 CSX4B6 14982951 IC50 = 720 nM T46360 C2SE6U 14982952 IC50 = 1800 nM T46360 CY3FM7 14982953 IC50 = 432 nM T46360 CC2HP8 14982954 IC50 = 165 nM T46360 CR8ZX1 14982955 IC50 = 227 nM T46360 CIG1W9 14982956 IC50 = 202 nM T46360 CNB0U1 14982957 IC50 = 297 nM T46360 CLG2A3 14982961 IC50 = 77 nM T46360 C83QWH 14982964 IC50 = 88 nM T46360 CJU87A 14982965 IC50 = 54 nM T46360 CJ2PE3 14982966 IC50 = 24 nM T46360 CY82JH 14982968 IC50 = 23 nM T46360 C59ETV 14982969 IC50 = 52 nM T46360 C8FHX4 14982970 IC50 = 100 nM T46360 CQV51D 14982971 IC50 = 237 nM T46360 CIFL16 14982976 IC50 = 80 nM T46360 CGE08Y 14982977 IC50 = 226 nM T46360 CR72BK 14982978 IC50 = 155 nM T46360 CIJ47C 14982979 IC50 = 164 nM T46360 COC5A3 14982980 IC50 = 53 nM T46360 C1Y4DM 14982981 IC50 = 1900 nM T46360 CODB98 14982982 IC50 = 49 nM T46360 C1Z9BL 14982983 IC50 = 347 nM T46360 CRF43C 14982984 IC50 = 2100 nM T46360 C3CXH1 14982992 IC50 = 33 nM T46360 C3BK0M 14982993 IC50 = 92 nM T46360 C0YQF8 14982994 IC50 = 45 nM T46360 C31OGY 14982995 IC50 = 16 nM T46360 CELY61 14982996 IC50 = 22 nM T46360 CU8X7Q 14982997 IC50 = 36 nM T46360 C89ZMJ 14983027 IC50 = 29 nM T46360 CJB9L5 14983028 IC50 = 119 nM T46360 CE2LO0 14983029 IC50 = 175 nM T46360 C7V0FZ 14983030 IC50 = 129 nM T46360 C8XK3F 14983031 IC50 = 320 nM T46360 C0F2YM 14983032 IC50 = 76 nM T46360 COHF72 14983033 IC50 = 194 nM T46360 CE62QX 14983034 IC50 = 164 nM T46360 C9XB8N 14983035 IC50 = 95 nM T46360 CT9B0C 14983036 IC50 = 493 nM T46360 CUD3A8 14983037 IC50 = 254 nM T46360 CE0OG6 14983038 IC50 = 159 nM T46360 CL0QW6 14983039 IC50 = 50 nM T46360 CV4XG6 14983040 IC50 = 51 nM T46360 CAD38J 14983041 IC50 = 190 nM T46360 C83IQA 14983042 IC50 = 46 nM T46360 CHMC30 14983043 IC50 = 84 nM T46360 C0E1GY 14983044 IC50 = 139 nM T46360 CG7SN0 14983045 IC50 = 95 nM T46360 CE2XK1 14983046 IC50 = 32 nM T46360 CW3R4M 14983047 IC50 = 63 nM T46360 C5YAV6 14983048 IC50 = 73 nM T46360 CY40QK 14983049 IC50 = 119 nM T46360 CMPN17 14983050 IC50 = 67 nM T46360 CHG9L5 14983053 IC50 = 34 nM T46360 CI79PE 14983054 IC50 = 26 nM T46360 CY1ZT7 14983055 IC50 = 93 nM T46360 C4X9RT 15034720 Ki = 41 nM T46360 C0JVK6 15034721 Ki = 34 nM T46360 C6FLJ0 15034722 Ki = 14 nM T46360 C1XUR9 15034723 Ki = 15 nM T46360 CYJ8D3 15034724 Ki = 19 nM T46360 C1E9DR 15034725 Ki = 18 nM T46360 C0CML8 15034727 Ki = 16 nM T46360 CRD98J 15034728 Ki = 62 nM T46360 CW97AB 15034729 Ki = 31 nM T46360 C7DE2A 15034730 Ki = 17 nM T46360 C0XTN3 15034731 Ki = 5 nM T46360 CU3V1E 15034733 Ki = 16 nM T46360 C3DIU6 15034734 Ki = 3 nM T46360 CF6BC5 15034735 Ki = 24 nM T46360 CSZ6G9 15034737 Ki = 15 nM T46360 C20NWP 15034738 Ki = 2 nM T46360 CU5I8Q 15034740 Ki = 250 nM T46360 CT91RK 15034743 Ki = 170 nM T46360 CGA52B 15034744 Ki = 19 nM T46360 CFQB36 15061885 Ki = 9.5 nM T46360 COQ0S2 15061886 Ki = 6.2 nM T46360 CE74WO 15061887 Ki = 3.4 nM T46360 C4R7ZN 15061888 Ki = 9.3 nM T46360 CSI1G0 15061889 Ki = 6.3 nM T46360 CI8CY0 15061890 Ki = 27.4 nM T46360 C7NR1V 15061896 Ki = 27.1 nM T46360 CG3T6K 15061897 Ki = 6 nM T46360 C4S2OB 15061898 Ki = 8.8 nM T46360 C6BJ0T 15061899 Ki = 12 nM T46360 CV8K6X 15061903 Ki = 83.2 nM T46360 CO31ZL 15061905 Ki = 7.9 nM T46360 CY1KZ4 15061906 Ki = 20 nM T46360 C6NL4F 15065448 IC50 = 17 nM T46360 C7R4WQ 15065449 IC50 = 7 nM T46360 C82EDI 15065450 IC50 = 7 nM T46360 CX7DC9 15065451 IC50 = 8 nM T46360 C61DXO 15065452 IC50 = 13 nM T46360 CYTG20 15065453 IC50 = 9 nM T46360 COBY80 15065454 IC50 = 3.2 nM T46360 CE35OQ 15065456 IC50 = 8 nM T46360 CAK96V 15113293 Ki = 1.76 nM T46360 CAL9M2 15113300 Ki = 5.78 nM T46360 C4H1NE 15113301 Ki = 277 nM T46360 CU7I0M 15113304 Ki = 1.35 nM T46360 COD14I 15113305 Ki = 11.7 nM T46360 CC4U7N 15113306 Ki = 0.84 nM T46360 CZ5XG0 15113307 Ki = 2.09 nM T46360 CQ26WU 15113308 Ki = 0.73 nM T46360 CN75UR 15113309 Ki = 20.18 nM T46360 CJO12C 15113311 Ki = 1.46 nM T46360 C8L6WJ 15113312 Ki = 0.62 nM T46360 C0BUH8 15113313 Ki = 0.38 nM T46360 CP7Z9O 15149381 IC50 = 116 nM T46360 C7ZQ8S 15149384 IC50 = 1612 nM T46360 C3ZK6U 15149386 IC50 = 474 nM T46360 CGBZ29 15149390 IC50 = 3560 nM T46360 CPZ2Q5 15149391 IC50 = 1276 nM T46360 CA10MG 15149392 IC50 = 1763 nM T46360 CR6HS1 15149393 IC50 = 2750 nM T46360 CZTR71 15149394 IC50 = 234 nM T46360 CR19PC 15149395 IC50 = 81 nM T46360 CK6CR7 15149396 IC50 = 348 nM T46360 CV5WQ2 15149397 IC50 = 534 nM T46360 CD1G7K 15149398 IC50 = 4876 nM T46360 CXB9C3 15149399 IC50 = 400 nM T46360 COK78H 15149400 IC50 = 262 nM T46360 C2NW3G 15149401 IC50 = 148 nM T46360 C8UCG2 15149402 IC50 = 88 nM T46360 C7KA2N 15149403 IC50 = 21 nM T46360 C1HR0I 15149404 IC50 = 105 nM T46360 C9KNO8 15149405 IC50 = 66 nM T46360 CW5MC6 15149406 IC50 = 129 nM T46360 CCH01D 15149407 IC50 = 133 nM T46360 CM2P4G 15149408 IC50 = 1483 nM T46360 CEWY20 15149409 IC50 = 702 nM T46360 CG7Q6W 15149411 IC50 = 1382 nM T46360 CX79WN 15149412 IC50 = 86 nM T46360 C6QL3P 15149413 IC50 = 3044 nM T46360 CHBC48 15149414 IC50 = 44 nM T46360 CN0P7T 15149415 IC50 = 8085 nM T46360 CAG3U8 15149416 IC50 = 836 nM T46360 CWN18O 15149417 IC50 = 85 nM T46360 CCH6M2 15149418 IC50 = 76 nM T46360 C8K5YO 15149419 IC50 = 231 nM T46360 CP83UL 15149420 IC50 = 267 nM T46360 C6O1FB 15149421 IC50 = 212 nM T46360 C7F1XV 15149422 IC50 = 482 nM T46360 CPE03W 15149426 IC50 = 3950 nM T46360 CV79PM 15163132 IC50 = 5.495 nM T46360 CG64QT 15163133 IC50 = 6.761 nM T46360 CSYU86 15163134 IC50 = 69.18 nM T46360 C20RCB 15163135 IC50 = 74.13 nM T46360 CM82BJ 15163136 IC50 = 6.761 nM T46360 CXWA38 15163138 IC50 = 4.786 nM T46360 CFMK89 15163140 IC50 = 1.047 nM T46360 CD4N5E 15163141 Ki = 0.6 nM T46360 C6JO1G 15163142 IC50 = 2.291 nM T46360 C4TX7I 15163143 IC50 = 2.884 nM T46360 CU3KS6 15163144 IC50 = 5.012 nM T46360 C8GZW1 15163145 IC50 = 6.607 nM T46360 CPIL08 15163146 IC50 = 10.23 nM T46360 CX3L5P 15163147 IC50 = 18.2 nM T46360 CI48UB 15163148 IC50 = 1.413 nM T46360 C9WFS6 15163149 IC50 = 1.66 nM T46360 CMZ73A 15163150 IC50 = 6.761 nM T46360 CTZ6J7 15163151 IC50 = 14.13 nM T46360 C1QZA4 15163152 IC50 = 9.55 nM T46360 C9V2LE 15163153 IC50 = 6.31 nM T46360 CEJ3H5 15163154 IC50 = 5.495 nM T46360 CAM8N1 15163155 IC50 = 11.22 nM T46360 C07FGX 15163160 IC50 = 1.349 nM T46360 C59BLX 15163161 IC50 = 1.514 nM T46360 C1JY2C 15163162 IC50 = 2.042 nM T46360 C36LSH 15163163 IC50 = 3.467 nM T46360 CGW2U3 15163164 IC50 = 3.162 nM T46360 CT0FG7 15163165 IC50 = 16.22 nM T46360 CKQL79 15166841 Ki = 2.72 nM T46360 CLIK54 15166843 Ki = 44.5 nM T46360 CL25QN 15166844 Ki = 10.3 nM T46360 CRX06M 15166845 Ki = 2.13 nM T46360 CA58OD 15175719 Ki = 1.19 nM T46360 C6EQD1 15175722 Ki = 0.54 nM T46360 CB0M5G 15205702 Ki = 46.5 nM T46360 C2B9YF 15205887 Ki = 1200 nM T46360 CX8YP7 15229597 Ki = 7 nM T46360 C4XSK7 15230909 IC50 = 100 nM T46360 CCZ8K3 15288693 Ki = 3 nM T46360 CWJ12B 15340879 Ki = 3 nM T46360 CR4UB7 15379806 IC50 = 26 nM T46360 CFQU06 15379808 IC50 = 16 nM T46360 CXP2Q0 15428989 Ki = 1.4 nM T46360 CZ72SA 15489265 Ki = 78.7 nM T46360 C65SCN 15599151 Ki = 484 nM T46360 CD0ZG3 15601069 Ki = 5200 nM T46360 CW3U0L 15646123 IC50 = 1212 nM T46360 C7UMB1 15646135 IC50 = 25 nM T46360 C0CXT6 15646139 IC50 = 37 nM T46360 C37SJN 15646141 IC50 = 38 nM T46360 CF2G1M 15646180 IC50 = 54 nM T46360 CRYD49 15657191 IC50 = 3305 nM T46360 C9P8QD 15657199 IC50 = 16.98 nM T46360 C1D0AP 15657202 IC50 = 0.2884 nM T46360 CSI49R 15657205 IC50 > 10000 nM T46360 C47CMD 15657207 IC50 = 10.47 nM T46360 C3E1TB 15657209 IC50 = 79.43 nM T46360 CUX59A 15657212 IC50 = 8.9 nM T46360 CG4LS3 15657214 IC50 = 117 nM T46360 C2F1JU 15657216 IC50 = 26.5 nM T46360 C12MGR 15657218 IC50 = 2.239 nM T46360 C5YG3C 15657219 IC50 = 3342 nM T46360 C57CUI 15701658 Ki = 146 nM T46360 CIUE86 15701660 Ki = 55.7 nM T46360 C4RX3J 15701661 Ki = 140 nM T46360 C1AYL6 15701662 Ki = 3.5 nM T46360 CU96AV 15701663 Ki = 3.1 nM T46360 CGEF49 15701664 Ki = 38 nM T46360 C1U5HG 15701665 Ki = 412 nM T46360 C1YFB9 15723883 Ki = 2.6 nM T46360 CDB0N6 15723885 Ki = 5.4 nM T46360 CVG95S 15723887 Ki = 2.8 nM T46360 CLN2V3 15723888 Ki = 125 nM T46360 C0JN7F 15723897 Ki = 4 nM T46360 CS98BY 15729885 IC50 = 23 nM T46360 C5NQL7 15729886 IC50 = 51 nM T46360 C6IFV4 15729897 IC50 = 1520 nM T46360 CU0J4B 15729898 IC50 > 45 nM T46360 C18DGR 15729900 IC50 = 12 nM T46360 C6ACS9 15729901 IC50 = 88 nM T46360 CJA86K 15729905 IC50 = 213 nM T46360 COLX61 15729907 IC50 = 504 nM T46360 CN95AB 15729914 IC50 = 227 nM T46360 CP7E8U 15729917 IC50 = 215 nM T46360 C7BH5E 15729921 IC50 > 1 nM T46360 CE87JV 15729922 IC50 = 3500 nM T46360 CG6FM7 15729925 IC50 > 2 nM T46360 C2LK6I 15729927 IC50 = 52 nM T46360 C7JK2U 15751758 IC50 = 3467.37 nM T46360 C9WX1R 15751761 IC50 = 1174.9 nM T46360 CE4TS7 15751762 IC50 = 338.84 nM T46360 C2CY5H 15751763 IC50 = 6.31 nM T46360 CMR8Q4 15751764 IC50 = 3.09 nM T46360 C40GZI 15751790 IC50 = 1.862 nM T46360 CZ69AV 15751791 IC50 = 3.981 nM T46360 C3QXB0 15751793 IC50 = 2.138 nM T46360 C4N9EK 15751794 IC50 = 1.413 nM T46360 CHL8I9 15767674 Ki = 1.57 nM T46360 C7JVH8 15767675 Ki = 82.5 nM T46360 CYCG42 15767676 Ki = 18.4 nM T46360 C45ITA 15767677 Ki = 5.68 nM T46360 C7H0OA 15767678 Ki = 1.47 nM T46360 CWH7G0 15767679 Ki = 1.75 nM T46360 CGF67P 15767680 Ki = 10.4 nM T46360 C7CLQ9 15767681 Ki = 3.81 nM T46360 CFH51J 15767682 Ki = 7.16 nM T46360 CR3LW7 15767683 Ki = 18.5 nM T46360 CFMC10 15767684 Ki = 130.6 nM T46360 CCP96Z 15767685 Ki = 4.68 nM T46360 CG8KR9 16005860 IC50 < 20 nM T46360 CAUP23 16048564 Ki = 2.2 nM T46360 C10CLM 16061352 Ki = 207 nM T46360 CTME96 16202156 Ki = 2150 nM T46360 CZ2IS9 16660294 Ki > 10000 nM T46360 CBH0C8 16664364 Ki = 2.1 nM T46360 CSNM61 16730082 Ki = 36.8 nM T46360 C0LEG4 17159068 Ki = 16 nM T46360 CA6E9Q 17159204 Ki = 2.5 nM T46360 C8O7EW 17176477 Ki = 15 nM T46360 C45JHX 17644936 Ki > 100 nM T46360 C7MST8 17758676 Ki = 3450 nM T46360 CM36GJ 17867053 Ki = 8 nM T46360 C21FJV 17867054 Ki = 5 nM T46360 CCM1L3 18118650 Ki = 10 nM T46360 CZ31UL 18118651 Ki = 37 nM T46360 C9UE6C 18118654 Ki = 40 nM T46360 C30VIU 18703006 Ki = 0.76 nM T46360 CD4BH5 18703016 Ki = 0.17 nM T46360 C6D5UW 18790190 Ki = 0.38 nM T46360 CBY3Q2 18790194 Ki = 0.28 nM T46360 CWY32U 18790196 Ki = 0.19 nM T46360 CFYK37 18790204 Ki = 4.1 nM T46360 CXA1F2 18790208 Ki = 0.81 nM T46360 C04TCD 18790215 Ki = 190 nM T46360 C53XYC 18790234 Ki = 0.26 nM T46360 CCU7M5 18790248 Ki = 2.3 nM T46360 C2A7IW 18790250 Ki = 6.8 nM T46360 C71TDI 18790258 Ki = 0.29 nM T46360 CT8Y7L 18790272 Ki = 0.32 nM T46360 CF50XE 18790283 Ki = 1.5 nM T46360 C8W2PU 18959700 IC50 = 210 nM T46360 CZY57S 18959702 IC50 = 54 nM T46360 CX3BD8 18959714 IC50 = 58 nM T46360 CZFE27 18959715 IC50 = 118 nM T46360 C7Y2PB 18959716 IC50 = 263 nM T46360 C7Q1KM 18959727 IC50 = 91 nM T46360 C60MOL 18959733 IC50 = 195 nM T46360 CKUS01 18959739 IC50 = 54 nM T46360 CW8PK0 19022852 Ki = 5 nM T46360 COZ07Y 19093638 IC50 = 7.586 nM T46360 CS7A4F 19427051 IC50 = 72 nM T46360 C9KH6O 19427053 IC50 = 9 nM T46360 C4MGT6 19427060 IC50 = 6 nM T46360 C4T9LZ 19606389 IC50 = 210 nM T46360 C1YXZ6 20068647 IC50 > 49 nM T46360 CLH0Z3 20068655 IC50 = 89 nM T46360 C40JIT 21474204 Ki = 5 nM T46360 CRT1Q8 21481466 Ki = 17 nM T46360 C3T5HF 21509921 Ki = 6143 nM T46360 CT7XG9 21830793 Ki = 59 nM T46360 CD5ZM4 21846520 Ki = 74 nM T46360 C2PEQ0 21968329 Ki = 45 nM T46360 CYM17I 22024852 Ki = 9.6 nM T46360 C1I4MZ 22413499 Ki = 2 nM T46360 CVGW27 22875688 Ki = 1.08 nM T46360 CIL6K7 22875693 Ki = 2.53 nM T46360 C72YBR 22875695 Ki = 1.2 nM T46360 C6E2DA 23465639 Ki = 0.06607 nM T46360 CYE83W 24739748 Ki = 233 nM T46360 CP9LR1 24739752 Ki = 128 nM T46360 CDN32O 24743568 Ki = 39 nM T46360 C6B2QL 24743571 Ki = 80.8 nM T46360 C54VFU 24743572 Ki = 9.5 nM T46360 CC52AB 24743739 Ki = 7.2 nM T46360 C5WGF4 24744816 Ki > 1000 nM T46360 C1SDO5 24744977 Ki = 23.1 nM T46360 CC36WF 24835442 Ki = 9 nM T46360 CDC91N 24839550 Ki = 100 nM T46360 CBGO31 24867245 Ki = 1.8 nM T46360 CET2U8 25005670 IC50 = 3.2 nM T46360 CDZ67U 25006418 IC50 = 48.1 nM T46360 C1OJ8G 25006786 IC50 = 2.9 nM T46360 CWT7P6 25059251 Ki = 2.9 nM T46360 CD7SE4 25060019 Ki = 24 nM T46360 CA1EJ2 25120700 Ki = 392 nM T46360 C1SH4X 25167085 Ki = 4.5 nM T46360 CX7QS0 25167087 Ki = 2.1 nM T46360 C90IWB 25184808 Ki = 5484 nM T46360 CWQ5S7 27148262 Ki = 4.3 nM T46360 C4MRQ0 27842480 Ki = 383 nM T46360 CUVS17 29048070 Ki = 2.9 nM T46360 CNK45Q 29150590 Ki = 41 nM T46360 C85BLI 30675158 Ki = 21 nM T46360 CR9N7G 30853613 Ki = 23 nM T46360 C7EJK2 31588412 Ki = 1.9 nM T46360 CO9HV7 40624141 Ki = 42 nM T46360 CRJ5E1 41306333 Ki = 47 nM T46360 CCF93H 41306385 Ki = 3.9 nM T46360 CQSO71 41306434 Ki = 24 nM T46360 CGO25K 41306445 Ki = 10 nM T46360 C83TBP 41307231 Ki = 2.9 nM T46360 CNY78F 42601649 IC50 = 954.99 nM T46360 CJH9I7 42601650 IC50 = 12.88 nM T46360 C7X6FE 42601651 IC50 = 4.467 nM T46360 CFB67A 42601652 IC50 = 58.88 nM T46360 C5J4MX 42601814 IC50 = 5.495 nM T46360 C8WNV1 42601815 IC50 = 17.38 nM T46360 CD81XZ 43267406 IC50 > 100000 nM T46360 CYI6L0 44248689 Ki > 100 nM T46360 CT1R7P 44270247 Ki = 100 nM T46360 C71EWU 44270248 Ki = 2000 nM T46360 C1CMA5 44272667 Ki = 17.7 nM T46360 C7ZMY2 44272754 Ki = 5.7 nM T46360 C5X7RV 44272941 Ki = 30 nM T46360 CBV83R 44272942 Ki = 0.9 nM T46360 C12IYN 44273058 Ki = 5.8 nM T46360 C8CEB5 44273063 Ki = 0.48 nM T46360 CU1HB5 44273339 Ki = 135 nM T46360 C6UN9B 44273356 Ki = 8.6 nM T46360 CQ35UT 44273357 Ki = 19.4 nM T46360 CU71HE 44273383 Ki = 130 nM T46360 C1M4OC 44273461 Ki = 124 nM T46360 CBH0I3 44285300 IC50 = 928 nM T46360 C1MV9C 44285320 IC50 = 63 nM T46360 CVP97C 44285332 IC50 = 65 nM T46360 C4DZY7 44285419 IC50 = 130 nM T46360 CCD68A 44285462 IC50 = 16 nM T46360 CQ4U7F 44285482 Ki = 31.8 nM T46360 CK70ZR 44285702 IC50 = 1630 nM T46360 CWJ9C4 44285740 IC50 = 99 nM T46360 CTR39Y 44291865 Ki = 34 nM T46360 CG1AV3 44292277 Ki = 270 nM T46360 CRT6Q8 44292278 Ki = 300 nM T46360 CVHM52 44292312 Ki = 120 nM T46360 C6PZU2 44292354 Ki = 1 nM T46360 C4H6US 44296111 Ki = 115 nM T46360 CGM01C 44296419 Ki = 456 nM T46360 CT4OF7 44296433 Ki = 161 nM T46360 C6QL4P 44296593 Ki = 49 nM T46360 CM92GY 44296633 Ki = 245 nM T46360 CL5CV9 44296635 Ki = 49 nM T46360 CBGJ28 44296645 Ki > 3300 nM T46360 C7ICW0 44296647 Ki = 241 nM T46360 CWZ4L2 44296655 Ki = 14 nM T46360 C0CS2T 44296665 Ki > 3300 nM T46360 C9GE4U 44297117 Ki > 1000 nM T46360 CMY2U8 44298009 Ki = 8.3 nM T46360 CZL87E 44303090 Ki = 1.7 nM T46360 CTBP60 44303758 Ki = 28 nM T46360 CN5B1M 44304225 IC50 = 4.677 nM T46360 CZA85U 44304236 IC50 = 6.607 nM T46360 CPV5R8 44304238 IC50 = 7.079 nM T46360 CRQ62S 44304240 IC50 = 16.6 nM T46360 CZ9IE3 44304242 IC50 = 81.28 nM T46360 C5DZ7S 44304251 IC50 = 0.2512 nM T46360 C04AXY 44304253 IC50 = 1.175 nM T46360 CWK5I3 44304261 IC50 = 4.571 nM T46360 CRK8S1 44304359 IC50 = 1.738 nM T46360 CIMW61 44304370 IC50 = 2.042 nM T46360 CY9L8D 44304372 IC50 = 2.455 nM T46360 C97XJP 44304406 IC50 = 8.71 nM T46360 C83NIJ 44304409 IC50 = 97.72 nM T46360 C90SZX 44304411 IC50 = 1.995 nM T46360 CNW1J7 44304414 IC50 = 1.82 nM T46360 CF96TW 44304421 IC50 = 2.291 nM T46360 CH2IG4 44304429 IC50 = 2.188 nM T46360 CNS9U4 44304433 IC50 = 4.266 nM T46360 C64ZWJ 44304443 IC50 = 3.467 nM T46360 CEJ6O9 44304447 IC50 = 0.3236 nM T46360 C4BHF5 44304618 IC50 = 2.57 nM T46360 C8Z3WP 44307427 IC50 = 9 nM T46360 CGZ1J8 44307523 Ki = 1.78 nM T46360 C7PZH9 44309297 Ki = 19 nM T46360 COHQ97 44309298 Ki = 8.4 nM T46360 CB2HT7 44309448 Ki = 1140 nM T46360 CT1E5L 44309453 Ki = 6220 nM T46360 C9Y7AI 44309455 Ki = 4 nM T46360 C7HA6I 44309464 Ki = 695 nM T46360 CJN2V0 44309466 Ki = 26 nM T46360 C38TNP 44309468 Ki = 324 nM T46360 C74QMW 44309492 Ki = 4150 nM T46360 C70WAV 44309628 Ki = 5130 nM T46360 CGYQ08 44309667 Ki = 11 nM T46360 C1Q4JD 44309690 Ki = 462 nM T46360 C1MH5F 44309692 Ki = 35 nM T46360 CL3F0P 44309694 Ki = 30 nM T46360 CA98DZ 44309696 Ki = 24 nM T46360 C0QFX9 44309716 Ki = 12 nM T46360 CD8RJ0 44309721 Ki = 0.59 nM T46360 CDB5R0 44309737 Ki = 49 nM T46360 C3YF2M 44309781 Ki = 3 nM T46360 CX5DU2 44309807 Ki = 232 nM T46360 CN0CZ1 44309809 Ki = 4000 nM T46360 CMJ95H 44309824 Ki = 580 nM T46360 CV65SY 44309831 Ki = 17 nM T46360 CX8H4A 44309835 Ki = 384 nM T46360 CT8L0X 44309837 Ki = 32 nM T46360 CG97RP 44309852 Ki = 4520 nM T46360 CT37BP 44309854 Ki = 3500 nM T46360 CE2QW0 44309866 Ki = 8110 nM T46360 C51RVN 44309974 Ki = 223 nM T46360 CCQN61 44309978 Ki = 6 nM T46360 C4UZG0 44309993 Ki = 1 nM T46360 CLYS40 44309995 Ki = 1 nM T46360 CH86ST 44310013 Ki = 298 nM T46360 C9LHD4 44310018 Ki = 214 nM T46360 CUC5I7 44310027 Ki = 16 nM T46360 C03FIO 44310034 Ki = 44 nM T46360 CU0EA9 44310036 Ki = 16 nM T46360 CJYR45 44310038 Ki = 9 nM T46360 C7M5HP 44310050 Ki = 4 nM T46360 C09JTN 44310052 Ki = 4 nM T46360 C4MD0R 44310071 Ki = 2 nM T46360 CY6O4H 44310073 Ki = 1 nM T46360 CN19YU 44310110 Ki = 7500 nM T46360 CL8D2O 44310124 Ki = 90 nM T46360 C4FS9Q 44310126 Ki = 163 nM T46360 CKVO42 44310128 Ki = 20000 nM T46360 CI2TN6 44310145 Ki = 4 nM T46360 COQW09 44310585 Ki = 0.13 nM T46360 C6FM0E 44310664 Ki = 0.8 nM T46360 CRK70Y 44310683 Ki = 1.1 nM T46360 C56NHS 44310857 Ki = 0.66 nM T46360 CWX0S8 44310858 Ki = 0.48 nM T46360 C2VTJ3 44310861 Ki = 0.89 nM T46360 CN08YO 44310878 Ki = 1.3 nM T46360 C6L2KD 44310879 Ki = 1.4 nM T46360 CBVZ21 44310961 Ki = 1.9 nM T46360 C42QYO 44311177 Ki = 7300 nM T46360 C6BX5O 44311179 Ki = 30 nM T46360 C6HEB9 44311180 Ki = 7500 nM T46360 C02DAJ 44311195 Ki = 4 nM T46360 CH7Q9A 44311197 Ki = 5 nM T46360 CBZ06X 44311211 Ki = 1 nM T46360 C5YNX7 44311359 Ki = 1830 nM T46360 C6D5TP 44311361 Ki = 1590 nM T46360 C7VW2Z 44311445 Ki = 6880 nM T46360 C71HBP 44311480 Ki = 6 nM T46360 CRW2P1 44311482 Ki = 7 nM T46360 CCNT08 44311493 Ki = 352 nM T46360 CW8S4Z 44311613 Ki = 4 nM T46360 CO2P4D 44311615 Ki = 70 nM T46360 C3QI6S 44311621 Ki = 10 nM T46360 C9GN7W 44311623 Ki = 13 nM T46360 CTR73J 44311625 Ki = 34 nM T46360 C5IKM9 44311640 Ki = 131 nM T46360 CKMJ50 44312948 Ki = 64 nM T46360 C74HMA 44313623 Ki = 1.33 nM T46360 C3J7XK 44313729 Ki = 1.67 nM T46360 CP3IG8 44313766 Ki = 3 nM T46360 CUQ94M 44313811 Ki = 2.87 nM T46360 C6CTR9 44313813 Ki = 2.87 nM T46360 CYI1A5 44313950 Ki = 0.55 nM T46360 C09MRS 44314013 Ki = 9.04 nM T46360 C4YT2K 44314123 Ki = 1.7 nM T46360 CSX31U 44314127 Ki = 174 nM T46360 CR24KE 44314136 Ki = 1.6 nM T46360 CR2YW9 44314137 Ki = 78 nM T46360 CW79CE 44314138 Ki = 16.3 nM T46360 C8T6GO 44314139 Ki = 154 nM T46360 CIYN38 44314217 Ki = 80 nM T46360 C5DS0N 44314218 Ki = 607 nM T46360 CU27RC 44314387 Ki = 119 nM T46360 CH4R7E 44314603 Ki = 1.7 nM T46360 CJL61P 44315181 Ki = 90 nM T46360 CLCN19 44315510 Ki = 1 nM T46360 CC57FY 44315535 Ki = 5 nM T46360 CEU56A 44315536 Ki = 8 nM T46360 C2DB7M 44315537 Ki = 18 nM T46360 C06BLA 44315552 Ki = 4 nM T46360 CI9GC2 44315578 Ki = 212 nM T46360 CW2I9R 44315579 Ki = 28 nM T46360 CF3M9C 44315580 Ki = 12 nM T46360 CSF86X 44315581 Ki = 2 nM T46360 CJ78AN 44315794 Ki = 4 nM T46360 C6B4CM 44315795 Ki = 22 nM T46360 C2WNL8 44315815 Ki = 8 nM T46360 CMRY42 44315830 Ki = 18 nM T46360 CD5R0G 44318068 IC50 = 163 nM T46360 C9UI8D 44318072 IC50 = 120 nM T46360 CT8WG0 44319215 IC50 = 5312 nM T46360 C0IU3Z 44321002 Ki = 104 nM T46360 C7QE2P 44321166 Ki = 97.2 nM T46360 C0M8TC 44321369 Ki = 138 nM T46360 C45HNC 44321397 Ki = 124 nM T46360 C1M7CY 44321499 Ki = 4420 nM T46360 CD8W0B 44321533 Ki = 552 nM T46360 C1E7MU 44321569 Ki = 5720 nM T46360 CEC92Q 44321621 Ki = 11.1 nM T46360 CAUB15 44321622 Ki = 32.5 nM T46360 CQ5V8G 44321623 Ki = 29.6 nM T46360 C2IAK4 44321648 Ki = 596 nM T46360 CT7X9G 44327682 Ki = 5.86 nM T46360 C61RYB 44327700 Ki = 0.45 nM T46360 CP0OM3 44327701 Ki = 1.04 nM T46360 CLY6O9 44327702 Ki = 3.07 nM T46360 CR9K2G 44327733 Ki = 1.75 nM T46360 C7ECV6 44330983 Ki = 157 nM T46360 CA9YX4 44330991 Ki = 158.49 nM T46360 CNB74Y 44332157 Ki = 35.2 nM T46360 CG4HV0 44332382 Ki = 2.62 nM T46360 CT0C6R 44332389 Ki = 37.4 nM T46360 C52MIY 44332475 Ki = 70.6 nM T46360 C3QS4R 44332496 Ki = 120 nM T46360 CE9JG2 44332500 Ki = 231 nM T46360 CGF56B 44332508 Ki = 1.72 nM T46360 CG2BJ0 44332511 Ki = 71.5 nM T46360 C8L0CI 44332512 Ki = 68.6 nM T46360 CRW57S 44332515 Ki = 1.75 nM T46360 CIZ63N 44332579 Ki = 2.49 nM T46360 C3YHZ7 44334079 Ki = 64.9 nM T46360 C13AJE 44334211 Ki = 1.24 nM T46360 C26IAM 44336365 Ki = 21 nM T46360 CWQ04R 44336430 Ki = 300 nM T46360 C24UOF 44336449 Ki = 2090 nM T46360 C1UWR7 44337609 Ki = 5400 nM T46360 C26ITO 44340881 Ki = 2.6 nM T46360 CF94RB 44340893 Ki = 7 nM T46360 C6HED7 44340900 Ki = 5 nM T46360 CQ2M3C 44340915 Ki = 6 nM T46360 CXKI34 44340919 Ki = 4 nM T46360 CUW0O9 44340942 Ki = 8 nM T46360 CWZ0D7 44340945 Ki = 22 nM T46360 CP9J2Y 44341034 Ki = 1500 nM T46360 C1L8EB 44341173 Ki = 58 nM T46360 CK46JF 44341181 Ki = 5 nM T46360 CV62EA 44341349 Ki = 1.1 nM T46360 C4N6GE 44342597 Ki = 32 nM T46360 C0Z9DY 44342598 Ki = 35 nM T46360 CSZ34A 44342661 Ki = 49 nM T46360 CJVN97 44342684 Ki = 12 nM T46360 CP97HW 44342724 Ki = 1.9 nM T46360 C2EQZ1 44342741 Ki = 0.29 nM T46360 CYTQ61 44342743 Ki = 2.3 nM T46360 C0IJN7 44342746 Ki = 2.8 nM T46360 CQ5B8R 44342747 Ki = 38 nM T46360 CW5RB3 44342753 Ki = 1090 nM T46360 C1LQR9 44342754 Ki = 1330 nM T46360 CD3F2N 44342792 Ki = 6 nM T46360 CC1X5F 44342793 Ki = 43 nM T46360 C46PTB 44342843 Ki = 69 nM T46360 CNO76C 44342910 Ki = 18100 nM T46360 C5NQP9 44342911 Ki = 739 nM T46360 CNG79I 44342912 Ki = 45 nM T46360 CLC0Z1 44342925 Ki = 40 nM T46360 C74GDW 44342933 Ki = 104 nM T46360 CG1X6K 44342934 Ki = 16600 nM T46360 C2BPW6 44344745 IC50 = 182 nM T46360 CZV21Q 44347713 Ki = 26 nM T46360 CLG65Q 44347771 Ki = 5 nM T46360 CUI12W 44347787 Ki = 13 nM T46360 C7Q4IB 44347788 Ki = 174 nM T46360 CYP17T 44350537 Ki = 17.49 nM T46360 CD38RO 44350538 Ki = 117 nM T46360 C0K5CR 44350649 Ki = 95.69 nM T46360 CCU89V 44350664 Ki = 34.1 nM T46360 C3CM2E 44350704 Ki = 280.75 nM T46360 C03YVC 44350708 Ki = 249.3 nM T46360 CC3Y4A 44350710 Ki = 302.4 nM T46360 C8EF0H 44350786 Ki = 40.4 nM T46360 C5E3FK 44350787 Ki = 517.7 nM T46360 C41UID 44350800 Ki = 194.5 nM T46360 CRC5I3 44350810 Ki = 240.3 nM T46360 C69MTC 44350812 Ki = 191 nM T46360 CMRX47 44350817 Ki = 175 nM T46360 CZMW86 44350827 Ki = 30.89 nM T46360 CI7KH4 44350870 Ki = 380 nM T46360 C7NC0V 44350885 Ki = 106.8 nM T46360 C60IJH 44350886 Ki = 8.5 nM T46360 C4QP5U 44350942 Ki = 183 nM T46360 C50HVX 44350991 Ki = 32.5 nM T46360 C7FCG1 44351070 IC50 = 1250 nM T46360 C09PFU 44356418 IC50 = 3378 nM T46360 CMP3T6 44356420 IC50 = 130 nM T46360 CL0MH9 44356422 IC50 = 113 nM T46360 CR16SL 44356442 IC50 = 480 nM T46360 CNDC89 44356481 IC50 = 180 nM T46360 C3SZV2 44356483 IC50 = 178 nM T46360 C2GZ4I 44356488 IC50 = 224 nM T46360 CH53UR 44356504 IC50 = 494 nM T46360 C4U6DG 44356510 IC50 = 110 nM T46360 CD0G2I 44356520 IC50 = 112 nM T46360 C1E3PF 44356530 IC50 = 18.2 nM T46360 CBV4R6 44356532 IC50 = 113 nM T46360 CB0G7Y 44356538 IC50 = 221 nM T46360 CEZQ08 44356560 IC50 = 200 nM T46360 C4HJ1Q 44356562 IC50 = 40.2 nM T46360 CR3BG4 44356573 IC50 = 309 nM T46360 C9YHF4 44356579 IC50 = 4.5 nM T46360 C8NM9A 44356581 IC50 = 7.4 nM T46360 CL3EM6 44356583 IC50 = 5.7 nM T46360 CH0Z5S 44356587 IC50 = 45.3 nM T46360 CFUS27 44356589 IC50 = 205 nM T46360 C5W4TO 44356593 IC50 = 30.7 nM T46360 CU0M1F 44356607 IC50 = 15.8 nM T46360 C0IY2M 44356642 IC50 = 8 nM T46360 C5AM0K 44356750 IC50 = 203 nM T46360 CMQV74 44356752 IC50 = 261 nM T46360 CS4HR6 44356757 IC50 = 113 nM T46360 CL9H7O 44356759 IC50 = 1947 nM T46360 CYGJ56 44356761 IC50 = 79 nM T46360 CHRM80 44356783 IC50 = 115 nM T46360 CP1JG7 44356785 IC50 = 755 nM T46360 CE76RV 44356787 IC50 = 421 nM T46360 C8LI5Y 44356836 IC50 = 19.6 nM T46360 C8T9NZ 44356838 IC50 = 17.3 nM T46360 CVY7W0 44356840 IC50 = 23.9 nM T46360 CI2A0J 44357414 IC50 = 949 nM T46360 C35PQS 44357415 IC50 = 1830 nM T46360 CC7V3Q 44361163 Ki = 11.7 nM T46360 CT52YL 44361164 Ki = 31.7 nM T46360 C0XLF9 44361167 Ki = 14.8 nM T46360 CUB80P 44361281 Ki = 3.36 nM T46360 CY3F5S 44361297 Ki = 18.4 nM T46360 C4IZ6C 44361388 Ki = 5.74 nM T46360 CQOD63 44361659 IC50 = 8.5 nM T46360 C97MEH 44362252 Ki = 1.62 nM T46360 CE3KC6 44362800 Ki = 1.71 nM T46360 CHJI46 44364124 Ki = 3600 nM T46360 C6RHC8 44364145 Ki > 10000 nM T46360 CH93PJ 44364189 Ki = 1465 nM T46360 CEG3S1 44364199 Ki = 11.8 nM T46360 CRP3B1 44370359 Ki = 34.5 nM T46360 CF8TC4 44370527 Ki = 109 nM T46360 CCH1J0 44370541 Ki = 58.2 nM T46360 CYF19D 44378807 Ki = 18.6 nM T46360 C14WCF 44385319 IC50 = 9.7 nM T46360 CEY85C 44386517 Ki = 0.7 nM T46360 CX7W3K 44398003 Ki = 74 nM T46360 C2MZH9 44398036 Ki = 0.5 nM T46360 C7C2TW 44398114 Ki = 1 nM T46360 C17XVW 44398137 Ki > 100000 nM T46360 CM45OW 44398162 Ki = 5 nM T46360 C7E9FT 44403183 IC50 = 6.6 nM T46360 C08XKE 44403246 IC50 = 54 nM T46360 CI4J5V 44403247 IC50 = 77 nM T46360 CF6X3K 44460274 IC50 = 250 nM T46360 CZS51T 44460446 IC50 > 10000 nM T46360 CW0J1K 44573133 Ki = 2240 nM T46360 CC6GX9 44573260 Ki = 53 nM T46360 CWAX45 44573261 Ki = 1600 nM T46360 CU4X2D 44818602 Ki = 7.1 nM T46360 C4LOY2 45115589 Ki < 1000 nM T46360 CK5Z6Q 45160790 Ki = 1584.89 nM T46360 C69RIC 45260531 IC50 = 21.38 nM T46360 CEY5U0 45260638 Ki = 2.51 nM T46360 C4I6VA 45262124 IC50 = 82 nM T46360 CDB08V 45262186 IC50 = 30.1 nM T46360 CEYM15 45264502 IC50 = 16.6 nM T46360 C5H0TZ 45487178 Ki = 0.4365 nM T46360 C08PKX 45487184 Ki = 0.08913 nM T46360 CR46EI 45487199 Ki = 0.09772 nM T46360 C1KX4B 45487204 Ki = 0.05754 nM T46360 C4RCU0 45487212 Ki = 0.05248 nM T46360 CP8EI4 45487215 Ki = 0.1096 nM T46360 CT29RN 45489962 Ki = 3200 nM T46360 CKCN84 46225028 Ki = 2280 nM T46360 C34ZXM 46225029 Ki = 149 nM T46360 C46HRG 46877990 IC50 = 928 nM T46360 CN8QY1 46877991 IC50 = 1247 nM T46360 CFE82I 46877992 IC50 = 3650 nM T46360 CC3T9L 46877993 IC50 = 5303 nM T46360 CNW5M8 46877994 IC50 = 3267 nM T46360 CDYS63 46877995 IC50 = 42 nM T46360 CS1X3U 46877996 IC50 = 2670 nM T46360 C7M0RU 46877997 IC50 = 1335 nM T46360 CGN59L 46877998 IC50 = 200 nM T46360 CK5Z0C 46877999 IC50 = 228 nM T46360 C3JG1D 46878000 IC50 = 110 nM T46360 CJD01C 46878001 IC50 = 76 nM T46360 CRB5L6 46878002 IC50 = 870 nM T46360 CK7N6S 46878005 IC50 = 224 nM T46360 CYM6C0 46878006 IC50 = 1155 nM T46360 C85YUM 46878007 IC50 = 1609 nM T46360 CE72KC 46878008 IC50 = 302 nM T46360 CBG9X7 46878009 Ki = 11 nM T46360 CIN90O 46878010 IC50 = 196 nM T46360 CT1MY8 46878011 IC50 = 5952 nM T46360 CHV7E8 46878012 IC50 = 1385 nM T46360 CG98OY 46878013 IC50 = 211 nM T46360 C4T5FE 46878014 IC50 = 208 nM T46360 C3P1JH 46878015 IC50 = 2374 nM T46360 CWM1O2 46878220 Ki = 8554 nM T46360 CQ0J2T 46906592 Ki > 800 nM T46360 CPBM68 46906593 Ki > 800 nM T46360 CE9Y7S 46907276 Ki > 800 nM T46360 CID6G4 46907277 Ki > 800 nM T46360 C9L3ZI 46911069 Ki = 79.43 nM T46360 C1N4ID 49832807 Ki = 194 nM T46360 CWMU78 49853575 IC50 = 590 nM T46360 CLJK94 49853576 IC50 = 270 nM T46360 CC48YF 49853577 IC50 = 1200 nM T46360 CZ4B0R 49853579 IC50 = 210 nM T46360 C3C9EJ 49853580 IC50 > 100000 nM T46360 CTF02Q 49853581 IC50 = 7600 nM T46360 CN8JR2 49853583 IC50 = 15200 nM T46360 CK3S1W 49853672 IC50 = 11500 nM T46360 C98QPG 49853674 IC50 = 18800 nM T46360 CI4W2P 49853676 IC50 = 16300 nM T46360 CPI6N0 49853777 IC50 > 100000 nM T46360 C94GDK 49853778 IC50 > 100000 nM T46360 C85YTF 49853781 IC50 = 15800 nM T46360 CHV3U8 49853881 IC50 = 430 nM T46360 C7MGD9 49853882 IC50 = 7240 nM T46360 CTBY97 49853883 IC50 = 390 nM T46360 CQP63D 49853884 IC50 = 2250 nM T46360 CY8M9A 49853885 IC50 = 8410 nM T46360 CECY14 49853886 IC50 = 21100 nM T46360 CP6GK8 49853980 IC50 = 180 nM T46360 C0J1OX 49853981 IC50 > 100000 nM T46360 CJ0Q5W 49853983 IC50 = 11800 nM T46360 CHK26Y 49853984 IC50 = 930 nM T46360 CJWH91 49853986 IC50 = 18000 nM T46360 CN0JU9 49853987 IC50 = 500 nM T46360 C5OXM4 49854189 IC50 = 11600 nM T46360 C8DVX6 49855131 IC50 = 3250 nM T46360 CTV1K4 49855133 IC50 = 8830 nM T46360 C2RY0J 50878551 Ki = 302 nM T46360 C1W6TV 50898777 Ki = 398.11 nM T46360 CXMZ73 50898778 Ki > 10000 nM T46360 CU63SQ 50994498 Ki = 0.59 nM T46360 CE4KP1 51050257 Ki > 10000 nM T46360 C3A9OY 51111240 Ki = 20 nM T46360 CPJZ31 52149645 Ki = 5.8 nM T46360 C82HKM 52750322 Ki = 3.7 nM T46360 COCZ63 52912210 IC50 = 43 nM T46360 CMJ62D 53245590 Ki = 410 nM T46360 CMOZ61 53475319 Ki = 531 nM T46360 C4BWN0 53707349 Ki = 660 nM T46360 CWK70Q 54315083 Ki = 1640 nM T46360 CECV98 54581003 IC50 = 1.202 nM T46360 C7L9JS 54583594 Ki = 39 nM T46360 CWY64L 54591111 Ki = 83.4 nM T46360 C2Y7LX 54591112 Ki = 296 nM T46360 C3KO4E 56652775 Ki = 1492 nM T46360 CQ3SG5 56656039 Ki = 10320 nM T46360 CJKO58 56852956 Ki = 346.74 nM T46360 C1TC7Q 56963799 Ki > 10000 nM T46360 CXW2C4 57340967 Ki > 1000 nM T46360 CZU6L2 57345618 Ki = 2.884 nM T46360 CK9G8H 57345619 Ki = 3.6 nM T46360 C4EXS6 57396571 Ki = 51.7 nM T46360 CO3B4P 57399494 Ki = 63 nM T46360 CYN38R 57401819 Ki = 36 nM T46360 CZ2UB5 57705473 Ki = 14.2 nM T46360 C0JMC4 57861965 Ki = 879 nM T46360 C3TNQ5 60346448 Ki = 3.6 nM T46360 C7JG9R 60701380 Ki > 100 nM T46360 CW36YC 66561968 Ki = 10000 nM T46360 C7FMA4 70676458 Ki = 5090 nM T46360 CNL86E 70681422 IC50 = 63.3 nM T46360 C5IN6M 70683538 IC50 = 12.4 nM T46360 CNB3C9 70691984 IC50 > 100 nM T46360 C57VRM 70695522 IC50 = 299 nM T46360 C08PHA 70696149 IC50 = 0.27 nM T46360 CUD40A 70697541 IC50 = 9 nM T46360 CR5KY1 71061607 Ki > 5000 nM T46360 C72XPZ 71061659 Ki > 5000 nM T46360 CD1ET2 71061756 Ki > 5000 nM T46360 C5KM2W 71061887 Ki > 5000 nM T46360 CN7C9S 71222835 Ki = 29 nM T46360 C8QWT7 71222908 Ki = 58 nM T46360 C3HSF6 71222985 Ki = 18 nM T46360 C8SDY4 71222995 Ki = 98 nM T46360 CO3PG8 71223000 Ki = 16 nM T46360 CA6KM2 71223037 Ki = 141 nM T46360 CA8NH6 71223095 Ki = 514 nM T46360 CU64JP 71223100 Ki = 55 nM T46360 CN97QC 71223119 Ki = 399 nM T46360 CTC30W 71223161 Ki = 62 nM T46360 CO47LV 71223168 Ki = 371 nM T46360 CY17ZB 71223185 Ki = 116 nM T46360 CY9S4C 71223204 Ki = 11 nM T46360 CA03HG 71223206 Ki = 192 nM T46360 C7YJT8 71223208 Ki = 9 nM T46360 C89SAL 71223232 Ki = 156 nM T46360 C20GSJ 71223247 Ki = 25 nM T46360 CDP92M 71223250 Ki = 41 nM T46360 CGO4J3 71223252 Ki = 51 nM T46360 CFZ29E 71223262 Ki = 79 nM T46360 CW2D8E 71223267 Ki = 9 nM T46360 CEIG57 71223275 Ki = 32731 nM T46360 CU49ST 71223296 Ki = 23 nM T46360 CO19CM 71223298 Ki = 181 nM T46360 CS39DP 71223393 Ki = 716 nM T46360 CIMT57 71223397 Ki = 33 nM T46360 C8YB9W 71223407 Ki = 818 nM T46360 C02UWQ 71223427 Ki = 292 nM T46360 C3XTM8 71223439 Ki = 24 nM T46360 CLN1Q4 71223454 Ki = 119 nM T46360 CZR75D 71223459 Ki = 21 nM T46360 CY5K3O 71223493 Ki > 1000 nM T46360 C0W4UT 71223519 Ki = 100 nM T46360 C7KZ9O 71225558 Ki = 740 nM T46360 CL3E7G 71225577 Ki = 45 nM T46360 CDG9F6 71225600 Ki = 42923 nM T46360 C90WEH 71225643 Ki = 165 nM T46360 C32CRY 71225858 Ki = 6194 nM T46360 CW6IJ4 71225871 Ki = 200 nM T46360 CUYA72 71225882 Ki = 85 nM T46360 C3A5GS 71225888 Ki = 813 nM T46360 C47ZXI 71225920 Ki = 184 nM T46360 C7R0VL 71225947 Ki = 12 nM T46360 C2ZP6M 71225970 Ki = 946 nM T46360 CP9N6I 71225996 Ki = 294 nM T46360 C8B4HC 71226084 Ki = 13803 nM T46360 C8Y9VF 71226102 Ki = 112 nM T46360 CXG39S 71226177 Ki = 25770 nM T46360 C5MX6Z 71226198 Ki = 18000 nM T46360 CDTW51 71226340 Ki = 108 nM T46360 COY7Z0 71231455 Ki = 55 nM T46360 CCO7J6 71449812 Ki = 99.1 nM T46360 CDP7T0 71449813 Ki = 44 nM T46360 CXO90E 71449814 Ki = 139 nM T46360 CE3SF8 71449822 Ki = 8.9 nM T46360 CYLG97 71451628 Ki = 8.6 nM T46360 C3IN7Y 71451629 Ki = 13.3 nM T46360 CYG43C 71451630 Ki = 9.4 nM T46360 COL29E 71451631 Ki = 8.4 nM T46360 C0OBW8 71451632 Ki = 14.8 nM T46360 C2ENG0 71451633 Ki = 8.5 nM T46360 C4TWS5 71452172 Ki = 4.1 nM T46360 C26HJP 71452705 IC50 = 897 nM T46360 CPU9L0 71453455 Ki > 1000 nM T46360 C29CJD 71453456 Ki = 17.8 nM T46360 CG72SV 71453464 Ki = 16.5 nM T46360 C2IZQ3 71454076 IC50 = 12.3 nM T46360 CW3K2A 71455165 Ki = 65 nM T46360 CZ4HI3 71455166 Ki = 33.8 nM T46360 CMYL95 71455809 IC50 = 36.1 nM T46360 CE5K0Q 71456164 Ki = 762.3 nM T46360 CD0X6R 71456959 Ki > 1000 nM T46360 C4ZW0F 71457595 IC50 = 5.2 nM T46360 C1YGK5 71459491 IC50 = 2.9 nM T46360 CF8TR1 71459493 IC50 = 42 nM T46360 COE9Z8 71460635 Ki = 180 nM T46360 CZH53R 71460636 Ki = 33.3 nM T46360 C96HIW 71460640 Ki = 16.1 nM T46360 C2W9ZQ 71462356 Ki = 18.9 nM T46360 CK40DZ 71462357 Ki = 9.6 nM T46360 C0KR7M 71487770 Ki = 9 nM T46360 C63XQF 71487772 Ki = 22 nM T46360 CGB8N6 71488612 Ki = 13 nM T46360 C91OQB 71503148 Ki = 7 nM T46360 CK54BX 71601215 Ki = 1250 nM T46360 CBO95T 71601216 Ki = 1700000 nM T46360 C2S4EK 71654693 Ki = 536 nM T46360 CJ1S3B 71654694 Ki = 317 nM T46360 CGB32Z 71654695 Ki = 15 nM T46360 C6ZV8T 71655284 Ki = 194 nM T46360 CRFG67 71655285 Ki > 1000 nM T46360 CPOU74 71655286 Ki = 377 nM T46360 C29WRX 71655287 Ki > 1000 nM T46360 CQ70ER 71655288 Ki > 1000 nM T46360 CPW26Z 71655347 Ki = 79 nM T46360 CT8J6R 71655349 Ki > 1000 nM T46360 C0M8WK 71655351 Ki > 1000 nM T46360 CS31VA 71655413 Ki = 19 nM T46360 C0JQL7 71655415 Ki > 1000 nM T46360 CELM32 71655416 Ki = 178 nM T46360 CX72JE 71655418 Ki = 14 nM T46360 C8YHC4 71655477 Ki > 1000 nM T46360 CUHP20 71655478 Ki > 1000 nM T46360 CCD58E 71655480 Ki > 1000 nM T46360 CQIT18 71655541 Ki > 1000 nM T46360 CZN13Q 71655543 Ki > 1000 nM T46360 C94IXE 71655545 Ki > 1000 nM T46360 C7GP2C 71655610 Ki = 302 nM T46360 CL89HF 71655612 Ki = 245 nM T46360 CD78YO 71655614 Ki > 1000 nM T46360 CF78EW 71655616 Ki = 108 nM T46360 C9JF3X 71655681 Ki = 410 nM T46360 CVL20F 71655683 Ki = 67 nM T46360 CF9G8Q 71655685 Ki > 1000 nM T46360 CJ14RU 71655744 Ki > 1000 nM T46360 C6XU2K 71655746 Ki = 124 nM T46360 CDL35U 71655748 Ki = 30 nM T46360 CD63JO 71716506 Ki > 1000 nM T46360 C9M1OY 71716507 Ki = 6.3 nM T46360 CI3OB7 71717119 Ki = 2.75 nM T46360 CWOC31 71718342 Ki > 1000 nM T46360 CDN18F 72950534 Ki = 46.08 nM T46360 C8R1CQ 72950535 Ki = 13.36 nM T46360 C62XVD 72950697 Ki = 45.32 nM T46360 CJZW17 72950698 Ki = 38 nM T46360 CBV3X0 72950699 Ki > 1000 nM T46360 CX93FC 73056461 Ki = 34 nM T46360 CGDH92 73056753 Ki = 29 nM T46360 CC65OA 73213195 Ki > 10000 nM T46360 CW83DK 73213196 Ki = 218.78 nM T46360 CO79PJ 73345319 Ki = 40 nM T46360 CCV91B 73346042 Ki > 10000 nM T46360 C36ZPL 73350500 IC50 = 15200 nM T46360 C5X6WV 73353481 IC50 = 86800 nM T46360 CNA59Q 73354414 Ki = 38.9 nM T46360 C6P0HF 74766963 Ki = 100 nM T46360 CWK67L 74766964 Ki = 74 nM T46360 CWI54G 74766966 Ki = 82 nM T46360 C43THL 74766967 Ki = 732 nM T46360 C42MEP 74767042 Ki = 72 nM T46360 C9F2RU 74767046 Ki = 707 nM T46360 C1S8MT 74767047 Ki = 40.74 nM T46360 C6EX3U 74767048 Ki = 112 nM T46360 CAE45U 74767050 Ki = 666 nM T46360 CK3B4H 74767125 Ki = 300 nM T46360 CS2R9T 74767126 Ki = 95 nM T46360 CJ1W9E 74767127 Ki = 531 nM T46360 CPD9C5 74767128 Ki = 137 nM T46360 CV6KE8 74767129 Ki = 558 nM T46360 C7YR5T 74767130 Ki = 447 nM T46360 CI1GQ0 74767131 Ki = 926 nM T46360 CXLO16 74767207 Ki = 35 nM T46360 CK7WU2 74767208 Ki = 43 nM T46360 C98KAZ 74767209 Ki = 709 nM T46360 CE7RM5 74767211 Ki = 802 nM T46360 CX13JM 74767212 Ki = 31 nM T46360 C94IPS 74767213 Ki = 63 nM T46360 CAY81N 74767285 Ki = 31 nM T46360 C2SR1H 74767286 Ki = 39 nM T46360 C3FVE7 74767287 Ki = 48 nM T46360 C8RV5C 74767288 Ki = 11843 nM T46360 CVLI72 74767289 Ki = 9460 nM T46360 C7CIB1 74767290 Ki = 23832 nM T46360 CDA4B3 74767291 Ki = 1834 nM T46360 C0VXI7 74767363 Ki = 76 nM T46360 C4DEJ0 74767364 Ki = 475 nM T46360 CP92AE 74767365 Ki = 2915 nM T46360 CI61EO 74767366 Ki = 125 nM T46360 CY3AM9 74767367 Ki = 93 nM T46360 CK14JY 74767368 Ki = 1717 nM T46360 C8HA0F 74767448 Ki = 715 nM T46360 C2E7QW 75201901 Ki = 8200 nM T46360 CQ71AT 76073628 Ki = 5 nM T46360 C3AD4C 76313525 Ki = 0.91 nM T46360 C28RIZ 76518514 Ki = 21.88 nM T46360 CQ3EY1 76683576 Ki = 818 nM T46360 C5PW6K 76683678 Ki = 49 nM T46360 CXM51U 76683680 Ki = 31 nM T46360 CGE15Z 76683773 Ki = 46 nM T46360 CL03DO 76683775 Ki = 97 nM T46360 C8HAR3 76683777 Ki = 61 nM T46360 C1EY3H 76683779 Ki > 1000 nM T46360 CG0TR9 76683781 Ki = 10 nM T46360 C3O2FD 76683785 Ki = 781 nM T46360 C95OWP 76683875 Ki = 9 nM T46360 C01RIY 76683877 Ki = 12 nM T46360 C7SN9G 76683881 Ki = 9616 nM T46360 C67SLP 76683883 Ki = 23 nM T46360 C6IS1X 76683885 Ki = 52 nM T46360 CBSD29 76683976 Ki = 35 nM T46360 C1W4ER 76683978 Ki = 701 nM T46360 CITA80 76683982 Ki = 194 nM T46360 CC5J3B 76683988 Ki = 56 nM T46360 C0WR4O 76684092 Ki = 36 nM T46360 CJ1KN0 76684094 Ki = 13 nM T46360 C2XSM8 76684096 Ki = 878 nM T46360 CR76SA 76684100 Ki = 33 nM T46360 CLD49W 76684104 Ki = 62 nM T46360 C08EZV 76684202 Ki = 46 nM T46360 CGBP93 76684204 Ki > 1000 nM T46360 C75VCS 76684206 Ki = 70 nM T46360 CKC14S 76684208 Ki = 105 nM T46360 CV62NT 76684214 Ki = 58 nM T46360 CXO78M 76684294 Ki = 144 nM T46360 C8P7EC 76684296 Ki = 31 nM T46360 CG6C3U 76684304 Ki = 275 nM T46360 C1EF6U 76684306 Ki = 459 nM T46360 CB95UF 76684383 Ki = 388 nM T46360 C6MSH2 76684391 Ki = 111 nM T46360 C5VNK9 76684473 Ki > 1000 nM T46360 C2EO6P 76684475 Ki = 451 nM T46360 CI21ES 76684477 Ki = 216 nM T46360 COY67V 76684479 Ki = 241 nM T46360 CC81FG 76684481 Ki = 273 nM T46360 CI6K1G 76684564 Ki = 508 nM T46360 CLR0B8 78043801 Ki = 15 nM T46360 CZ75NQ 86582973 Ki = 51 nM T46360 CC0IB7 90146004 Ki = 112 nM T46360 CKH16N 90146246 Ki = 634 nM T46360 CY14OV 90269112 Ki = 662 nM T46360 C68URF 90269115 Ki > 1000 nM T46360 CM90FD 90643603 Ki = 7463 nM T46360 C5B8PY 90643604 Ki = 3063 nM T46360 CPN65E 90643787 IC50 = 30000 nM T46360 CLM0J5 90644067 Ki = 1148 nM T46360 CG83SL 90654976 Ki = 10 nM T46360 C4UEJ8 90654977 Ki = 3063 nM T46360 C5O4JQ 90654978 Ki = 10.5 nM T46360 C5IE8A 90655529 Ki = 29 nM T46360 C2SMQ1 90655530 Ki = 7.5 nM T46360 C7QRC3 90655531 Ki = 6.8 nM T46360 CK8M5I 90655532 Ki = 27 nM T46360 CZVJ18 90655533 Ki = 279 nM T46360 C1PAN6 90655534 Ki = 107 nM T46360 CU8FY3 90655535 Ki = 711 nM T46360 C6KXQ7 90655536 Ki = 465 nM T46360 CI35AY 90655537 Ki = 491 nM T46360 C8TOW0 90666080 Ki = 158.49 nM T46360 C2HF4P 90666081 Ki = 125.89 nM T46360 C1E9BD 90666082 Ki = 63.1 nM T46360 CH4Q1J 90666083 Ki = 63.1 nM T46360 COS08L 90666084 Ki = 1258.93 nM T46360 C1WUZ3 90666085 Ki = 398.11 nM T46360 CYUV14 90666086 Ki = 15.85 nM T46360 C9SMH8 90666087 Ki = 10 nM T46360 CZPD45 90666088 Ki = 25.12 nM T46360 CZX94Q 90666089 Ki = 630.96 nM T46360 C34WZM 90666090 Ki = 25.12 nM T46360 CT21RI 90666091 Ki = 199.53 nM T46360 CIBZ73 90666092 Ki = 100 nM T46360 CO7I5L 90666093 Ki = 79.43 nM T46360 CH5R8Q 98049507 Ki = 6300 nM T46360 C2EJK6 101910737 Ki = 1.1 nM T46360 CB5DK1 102004349 Ki = 6 nM T46360 CO6Z7J 110440208 Ki = 1.6 nM T46360 CBW0U9 110445832 Ki = 1.4 nM T46360 C5CDE0 118562359 Ki = 28 nM T46360 CS63OE 118562362 Ki = 209 nM T46360 CWH9B5 118562372 Ki = 91 nM T46360 C60BSA 118562375 Ki = 10 nM T46360 CE3D0A 118562384 Ki = 8 nM T46360 C7IVW9 118562402 Ki = 54 nM T46360 C63EGC 118562428 Ki = 53 nM T46360 CE53DJ 118562440 Ki = 8 nM T46360 CW26NV 118562451 Ki = 14 nM T46360 C7G5HO 118562469 Ki = 54 nM T46360 C3BIL8 118562502 Ki = 68 nM T46360 C5JKQ9 118562510 Ki = 6 nM T46360 C12CKV 118562522 Ki = 14 nM T46360 CF6LK7 118562538 Ki = 9 nM T46360 C6FOS9 118562556 Ki = 15 nM T46360 C25MXS 118562567 Ki = 11 nM T46360 C3TQE7 118562573 Ki = 88 nM T46360 CJF1E6 118562576 Ki = 40 nM T46360 C5QB2S 118562584 Ki = 21 nM T46360 C6TC3D 118562598 Ki = 53 nM T46360 CWA4B2 118562606 Ki = 13 nM T46360 C2EPN1 118565438 Ki = 99 nM T46360 C0XIN5 118567313 Ki = 32 nM T46360 C6PA1C 118567531 Ki = 103 nM T46360 CD4XK8 118567534 Ki = 14 nM T46360 CLVO18 118567538 Ki = 63 nM T46360 C1CP6Z 118567543 Ki = 58 nM T46360 C32PGF 118567545 Ki = 48 nM T46360 C7G8IT 118567547 Ki = 3 nM T46360 CN1DU3 118567549 Ki = 275 nM T46360 CKQ15C 118567550 Ki = 122 nM T46360 CJ43GO 118567552 Ki = 55 nM T46360 CV7U9Y 118567593 Ki = 237 nM T46360 CXW0K9 118567604 Ki = 11 nM T46360 C4ULH8 118567605 Ki = 13 nM T46360 C7DO6S 118567606 Ki = 13 nM T46360 C8TP7C 118567608 Ki = 8 nM T46360 C70RDE 118567618 Ki = 51 nM T46360 CGN3Z4 118567654 Ki = 26 nM T46360 CJOK48 118567670 Ki = 57 nM T46360 C4GDV1 118567672 Ki = 112 nM T46360 CK5T2Z 118567678 Ki > 1000 nM T46360 CCY60Z 118567689 Ki = 622 nM T46360 C59GUQ 118567742 Ki = 9 nM T46360 C36JSR 118567743 Ki = 8 nM T46360 C5NI2E 118567744 Ki = 38 nM T46360 CI0JY2 118567747 Ki = 39 nM T46360 CHU07G 118607283 Ki = 1.2 nM T46360 CX2QI6 118607309 Ki = 3.6 nM T46360 CIW02L 118607351 Ki = 4.3 nM T46360 C84QJX 118607364 Ki = 1.1 nM T46360 CX5B2A 118607439 Ki = 6.5 nM T46360 CXOT38 118607453 Ki = 7.3 nM T46360 C4U2GB 118607455 Ki = 1.7 nM T46360 CSB25E 118709750 Ki = 70.79 nM T46360 CD4S9R 118709751 Ki = 57 nM T46360 C4XS8G 118724294 Ki = 5.3 nM T46360 CG6O7M 118724295 Ki = 6.2 nM T46360 CLNB04 118724296 Ki = 4.3 nM T46360 CJ47XE 118724297 Ki = 18 nM T46360 CDL21J 118724298 Ki = 2 nM T46360 CT2RJ5 118724299 Ki > 200 nM T46360 C64SLY 118724300 Ki = 28 nM T46360 CK3RS5 118724301 Ki = 72 nM T46360 CC5E1Q 118724302 Ki = 160 nM T46360 CCE9F4 118724303 Ki = 7.2 nM T46360 CZC13F 118724304 Ki = 11 nM T46360 CQI71Z 118724305 Ki = 11 nM T46360 CJ1VY3 118724306 Ki = 2.5 nM T46360 C9ZR4V 118724307 Ki = 18 nM T46360 CR05GL 118724308 Ki = 11 nM T46360 CT36KB 118724309 Ki > 200 nM T46360 CTU50G 118724310 Ki = 36 nM T46360 CHP0Q2 118724311 Ki = 8 nM T46360 C5W8KO 118724312 Ki = 8.4 nM T46360 C8L5HP 118724313 Ki = 72 nM T46360 CHBZ37 118724314 Ki = 11 nM T46360 CYE4H7 118724315 Ki > 200 nM T46360 C1OHA6 118724316 Ki = 12 nM T46360 CTE58Z 118730369 Ki = 200 nM T46360 C3SL6R 118731566 Ki = 5.3 nM T46360 CSZ3F7 118731567 Ki = 1.2 nM T46360 C1TUD2 118731568 Ki = 0.9 nM T46360 C3NUS9 118731569 Ki = 6.4 nM T46360 C9WKE6 118731570 Ki = 10.3 nM T46360 CSZ4K3 118731571 Ki = 3.1 nM T46360 C1N6GY 118731572 Ki = 0.6 nM T46360 CMC9X4 118731573 Ki = 4.7 nM T46360 CL5H9N 118731574 Ki > 100 nM T46360 CSI32D 118731575 Ki = 2.2 nM T46360 CA8DB0 118731576 Ki > 100 nM T46360 CD01IE 118731577 Ki > 100 nM T46360 C5PXE8 118731578 Ki > 100 nM T46360 CNK9U1 118731579 Ki > 100 nM T46360 C8P6OB 118731580 Ki = 30.3 nM T46360 CT1G4C 118731581 Ki = 5.7 nM T46360 C6Q4SP 118731582 Ki > 100 nM T46360 CWE78H 118731583 Ki > 100 nM T46360 CH3TQ1 118732991 IC50 = 135 nM T46360 C7ODW3 122195524 Ki < 300 nM T46360 C5QIE8 124197459 Ki = 133 nM T46360 C09PAE 126744799 Ki = 205 nM T46360 COJ60B 126744800 Ki = 147 nM T46360 C2U4GO 126744949 Ki = 656 nM T46360 C0FKA4 126744972 Ki = 61 nM T46360 C79BZK 127026013 Ki = 31 nM T46360 C9E4NV 127026014 Ki = 2200 nM T46360 CTBN56 127026052 Ki = 85.11 nM T46360 C64OKQ 127027941 Ki = 676 nM T46360 CJ4YC0 127031397 Ki = 119 nM T46360 CBU9G2 127031398 Ki = 37 nM T46360 CE1IA7 127031399 Ki = 53 nM T46360 C4WKG9 127031403 Ki = 12 nM T46360 CEDM28 127031404 Ki = 130 nM T46360 CV5UH0 127031405 Ki = 350 nM T46360 CHN9X2 127031422 Ki = 124 nM T46360 C0CY9W 127031423 Ki = 57 nM T46360 CNH2V8 127031424 Ki = 13 nM T46360 C2W0HL 127031949 Ki = 122 nM T46360 CU49VE 127036186 Ki = 74.13 nM T46360 CG06BD 127036932 Ki = 97.72 nM T46360 CVW71O 127036953 Ki = 102.33 nM T46360 C9M5RN 127048369 Ki = 73 nM T46360 CLM5O3 127048370 Ki = 27 nM T46360 C6J3FW 127048371 Ki = 24 nM T46360 C1AX7T 127050366 Ki = 6 nM T46360 C8VKE5 127050367 Ki = 27 nM T46360 CH64PD 127050993 Ki = 2.4 nM T46360 C1UPC8 127050994 Ki = 2.8 nM T46360 CVH86Y 127050995 Ki = 1.6 nM T46360 CM3I6O 127051201 Ki = 6.4 nM T46360 C1CA7B 127051216 Ki = 2.2 nM T46360 C6L5ZK 127051267 Ki = 13 nM T46360 CB8W3Y 127051268 Ki = 7.2 nM T46360 CH3SP2 127051269 Ki = 38 nM T46360 CX3KP6 127051889 Ki = 3.2 nM T46360 C50GOC 130442480 Ki = 8000 nM T46360 CM04RF 130442572 Ki = 6900 nM T46360 CUD08L 134817200 Ki = 65.2 nM T46360 CZQS20 134828069 Ki = 5.7 nM T46360 CYB5V2 134828071 Ki = 5.1 nM T46360 CZ56GX 135423874 Ki = 743 nM T46360 CH96LU 135559170 Ki = 4000 nM T46360 C9C3LB 136056476 IC50 = 113 nM T46360 CN1I7A 137634153 Ki = 4200 nM T46360 CNH2K5 137639103 Ki = 2.3 nM T46360 C3Y8DJ 137643283 Ki = 2.6 nM T46360 CY56BC 137648624 Ki = 1.5 nM T46360 CU0OC3 137658890 Ki = 5.4 nM T46360 CC2DK4 137661600 Ki = 8.4 nM T46360 C1TQ2A 145953153 Ki = 6.5 nM T46360 CXEV63 145954849 Ki = 1418 nM T46360 CDGA65 145956728 Ki = 19 nM T46360 CZW93M 145979453 Ki = 99 nM T46360 CV43SZ 145980698 Ki = 57 nM T46360 C7H3GY 145986754 Ki = 38293 nM T46360 CC4KD9 145986903 Ki = 573 nM T46360 CS9R6C 145990153 Ki = 774 nM T46360 CC2G1V 146025727 Ki = 8800 nM T46360 CJA9T4 146597626 Ki = 15.85 nM T46360 C3D4UM 146597628 Ki > 10000 nM T46360 C7UHR0 146597630 Ki = 100 nM T46360 CCRS21 146597638 Ki > 10000 nM T46360 CM18OU 146597639 Ki = 2511.89 nM T46360 C42TIZ 146597651 Ki = 501.19 nM T46360 CL5PG8 146597666 Ki > 10000 nM T46360 C89YUC 146597677 Ki = 251.19 nM T46360 CU9G0O 146597678 Ki > 10000 nM T46360 C6TRC9 146641556 Ki = 316.23 nM T46360 C8I3YJ 146641558 Ki = 125.89 nM T46360 C3LBA0 146641564 Ki = 158.49 nM T46360 CFD4N9 146641568 Ki = 630.96 nM T46360 CP70WA 146641787 Ki = 251.19 nM T46360 C0WU5Y 146641788 Ki = 199.53 nM T46360 C10LOP 146641795 Ki > 10000 nM T46360 CG97ER 146709966 Ki = 3162.28 nM T46360 C6FX4M 147636204 Ki > 10000 nM T46360 CW4S2X 147652368 Ki > 10000 nM T46360 CF5B2L 147653864 Ki = 501.19 nM T46360 C5PNX8 148302367 Ki = 12.59 nM T46360 C2E5HK 149396365 Ki = 7.943 nM T46360 C9T0PS 153061504 Ki = 1000 nM T46360 CF7J3M 153287535 Ki = 50.12 nM T46360 C72MVW 153287537 Ki > 10000 nM T46360 CAF36V 153287539 Ki = 12.59 nM T46360 C1FA0K 153287541 Ki = 50.12 nM T46360 CEQ69Z 153287542 Ki = 39.81 nM T46360 C9A7SV 153287550 Ki > 10000 nM T46360 C91KST 153287551 Ki > 10000 nM T46360 C6P3SR 153287553 Ki = 501.19 nM T46360 C3G5CJ 153287557 Ki = 158.49 nM T46360 CW31CT 153287566 Ki = 162.18 nM T46360 CYP86E 153287567 Ki = 251.19 nM T46360 CS73ZC 153287568 Ki = 63.1 nM T46360 CV9G7Z 153287572 Ki = 1000 nM T46360 CO85KL 153287574 Ki = 316.23 nM T46360 CCD9N1 155512086 Ki = 1790 nM T46360 CTV8R1 155512151 Ki = 626 nM T46360 CV35ZN 155513505 Ki = 690 nM T46360 C0LR8C 155517675 Ki = 5.1 nM T46360 C4KWA1 155518665 Ki = 113 nM T46360 C0IHP6 155518770 Ki = 25.7 nM T46360 CUSA24 155519891 Ki = 39.81 nM T46360 C9W2NV 155525645 Ki = 31.62 nM T46360 CP76JX 155526977 Ki = 398.11 nM T46360 CQT9R0 155527577 Ki = 77.62 nM T46360 CQV19C 155528829 Ki = 55 nM T46360 CPA51T 155528865 Ki = 95 nM T46360 CMNU06 155529976 Ki = 20.89 nM T46360 CS2MF5 155532495 Ki = 251.19 nM T46360 CB79ZW 155536080 Ki = 125.89 nM T46360 C5IK2Y 155536631 Ki = 22 nM T46360 CR16NT 155540848 Ki = 63 nM T46360 CI7FN8 155545740 Ki = 21 nM T46360 CIA1C9 155547197 Ki = 63 nM T46360 CF7MQ8 155550094 Ki = 630.96 nM T46360 C8AGX6 155550691 Ki = 5.1 nM T46360 CI41QF 155552117 Ki = 1970 nM T46360 CJ92EA 155552895 Ki = 501.19 nM T46360 CKSZ39 155553997 Ki = 6.9 nM T46360 C04OFL 155554079 Ki = 7.2 nM T46360 CRU26E 155554287 Ki = 39.81 nM T46360 C6ZWX1 155554837 Ki = 16 nM T46360 CZ9U5N 155554849 Ki = 316.23 nM T46360 CC48RQ 155556295 Ki = 148 nM T46360 CBS89O 155556618 Ki = 1500 nM T46360 CQ7Y5M 155556668 Ki = 4.9 nM T46360 CJBX01 155557042 Ki = 125.89 nM T46360 C4J0ZI 155559223 Ki = 199.53 nM T46360 C13RCK 155561279 Ki = 70 nM T46360 CXYQ73 155561471 Ki = 63.1 nM T46360 CCOD50 155562467 Ki = 3570 nM T46360 C6YO5L 155562543 Ki = 43.65 nM T46360 CK9RN6 155563452 Ki = 24.55 nM T46360 CSM7V1 155564110 Ki = 30 nM T46360 CP9TR0 10324985 Ki = 480 nM T46360 CEA0P3 12233037 Ki = 0.67 nM T46360 CYZI29 12233038 Ki = 36.5 nM T46360 D00FUO 4416 Ki = 30 nM T46360 D00GSD 25107716 Ki > 5000 nM T46360 D00KIK 398369 Ki = 674 nM T46360 D00NQV 5041 Ki = 82.1 nM T46360 D00VHW 11152527 Ki = 2.5 nM T46360 D00VKV 62751 IC50 = 2060 nM T46360 D01HTH 60839 IC50 = 2535 nM T46360 D02BXG 398415 Ki = 3170 nM T46360 D02EHL 398376 Ki = 1730 nM T46360 D02WJT 7333 Ki = 15 nM T46360 D03LDH 10758200 Ki = 0.3 nM T46360 D03TDN 1342 Ki = 2720 nM T46360 D03TNT 5753 Ki = 35600 nM T46360 D04FBZ 5284595 IC50 = 48 nM T46360 D04JJL 14771671 IC50 = 245 nM T46360 D04JZJ 2838196 Ki = 370 nM T46360 D04LWD 11336800 Ki = 1.4 nM T46360 D04ZMS 11773145 Ki = 3.38 nM T46360 D05CGI 11245709 Ki = 1.4 nM T46360 D05EQG 5265 IC50 = 954.99 nM T46360 D06FUV 5311189 Ki = 234 nM T46360 D06RFW 13781937 IC50 = 270 nM T46360 D07AAZ 82553 IC50 = 1000 nM T46360 D07BAH 32893 Ki = 46400 nM T46360 D07OOI 3456 IC50 = 17 nM T46360 D07TKE 15723894 Ki = 3 nM T46360 D09CGH 188914 Ki = 1.26 nM T46360 D09NSH 10810249 Ki = 257.04 nM T46360 D09RPR 16737207 Ki > 10000 nM T46360 D09TDI 6472 Ki = 15.5 nM T46360 D0A0GU 44247568 Ki = 17 nM T46360 D0B3WX 5475158 IC50 = 181.97 nM T46360 D0C1LI 53378764 Ki = 2.83 nM T46360 D0E8FG 14952700 Ki = 2710 nM T46360 D0FF6S 16038374 IC50 > 10000 nM T46360 D0J1AE 10708590 Ki = 2.6 nM T46360 D0J6JT 1355 Ki = 6150 nM T46360 D0KL1P 10474335 Ki = 5.3 nM T46360 D0M4RW 5281878 IC50 = 14.79 nM T46360 D0N8WR 10390222 Ki = 92 nM T46360 D0O3GF 1220 Ki > 2427 nM T46360 D0P0XA 197060 Ki = 9310 nM T46360 D0Q5PC 6468 IC50 = 560 nM T46360 D0Q7FM 15443 Ki = 342 nM T46360 D0R5WX 11220953 Ki = 4.8 nM T46360 D0T1GZ 408731 Ki = 11.3 nM T46360 D0U3PC 398365 Ki = 9170 nM T46360 D0V4RP 1346 Ki = 11200 nM T46360 D0V5HV 4296 Ki = 1340 nM T46360 D0W2YN 2760172 Ki = 550 nM T46360 D0X4RC 7096 Ki = 11440 nM T46360 D0X7BG 4679312 Ki > 1000 nM T46360 D0Y3DR 608630 Ki = 2890 nM T52790 D05ZWG 108147 Ki > 10000 nM T52790 D06TQR 76287260 IC50 = 21000 nM T52790 D0CB2B 23653789 Ki = 2.4 nM T52790 D0G2XE 6918468 IC50 = 87 nM T52790 D0K5HI 5311424 Ki = 144 nM T52790 D0XS4X 11527495 Ki = 0.07586 nM T52790 D0ZM5O 9884366 IC50 = 4900 nM T52790 D00VPT 6604009 Ki = 277 nM T52790 D02TKI 132846 IC50 > 1000 nM T52790 D02YWV 9953599 Ki = 0.3162 nM T52790 D03SXN 104943 IC50 > 10000 nM T52790 D04RCG 10327792 Ki = 0.631 nM T52790 D05WJQ 104974 IC50 = 0.13 nM T52790 D08WVA 9915372 IC50 = 3.981 nM T52790 D08ZBV 132837 IC50 > 5000 nM T52790 D0C9FF 9939040 IC50 = 5.5 nM T52790 D0IP6X 219077 Ki = 35.5 nM T52790 D0J3QU 44351946 Ki = 0.92 nM T52790 C97NZR 124003 EC50 = 78.1 nM T52790 C20AYU 153996 Ki = 1 nM T52790 CB1P6S 163828 IC50 = 2.5 nM T52790 CUIX42 190884 Ki = 1.445 nM T52790 C5N1KX 1760285 Ki = 237 nM T52790 CMLC05 1760287 Ki = 237 nM T52790 CZT46B 3570748 IC50 = 2.5 nM T52790 C0UR7K 4529080 Ki = 2947 nM T52790 C15UHN 5487475 Ki = 0.1549 nM T52790 C5PO1F 6604014 Ki = 1221 nM T52790 CE57YD 6604858 Ki = 1221 nM T52790 C36VYU 7016092 IC50 > 5000 nM T52790 C2W6PI 8867347 Ki = 12000 nM T52790 CPRQ41 9806459 Ki = 1 nM T52790 CYP28G 9807403 IC50 = 7.943 nM T52790 CL81MT 9809876 Ki = 67 nM T52790 CIGT19 9810434 Ki = 0.8 nM T52790 C35MSJ 9810544 Ki = 0.4 nM T52790 CP38OJ 9825316 Ki = 2.4 nM T52790 C5Q8EM 9828448 Ki = 9.2 nM T52790 CMJ7P3 9829402 Ki = 1.995 nM T52790 CR6CG0 9830304 IC50 = 24 nM T52790 C07FWV 9830361 Ki = 0.6 nM T52790 CN6WE9 9831075 Ki = 0.7 nM T52790 CZ2EY1 9831309 IC50 = 8.4 nM T52790 CR3XL0 9831504 Ki = 0.02512 nM T52790 C9BDV3 9831546 Ki = 0.2 nM T52790 CHIS10 9831674 Ki = 1.2 nM T52790 C3TV1U 9831707 Ki = 0.5 nM T52790 CU85VO 9832198 IC50 = 129 nM T52790 CZQ96M 9843958 IC50 = 22 nM T52790 C52PUJ 9849950 Ki = 18.5 nM T52790 C8MW2V 9849962 IC50 < 7 nM T52790 CC7P4X 9850582 Ki = 0.6 nM T52790 CIXG30 9852376 IC50 = 2.2 nM T52790 CMZ20K 9852630 Ki = 0.7 nM T52790 C2JS5O 9852904 Ki = 35 nM T52790 CSU2Y3 9853636 Ki = 0.5 nM T52790 CY37UT 9853827 Ki = 0.1585 nM T52790 C3LOJ7 9872857 Ki = 0.7 nM T52790 C2NP3I 9874027 Ki = 0.631 nM T52790 CM3O6E 9874168 IC50 = 18.8 nM T52790 CCE74U 9874473 Ki = 22 nM T52790 CD6U7Z 9875034 Ki = 0.4 nM T52790 CA2X8G 9875056 Ki = 0.8 nM T52790 CBT1R2 9887650 Ki = 7.943 nM T52790 CW07IY 9896757 Ki = 0.7 nM T52790 CF3M7Z 9914111 Ki = 3.5 nM T52790 CFP74K 9916195 IC50 = 6 nM T52790 C4SEJ2 9917970 Ki = 0.8 nM T52790 C5U0EO 9918479 Ki = 2.7 nM T52790 CH97DG 9939307 Ki = 1.6 nM T52790 CPZ4B5 9956370 Ki = 4.2 nM T52790 CQ69EA 9957749 Ki = 811 nM T52790 CMGB40 9959481 IC50 = 0.3981 nM T52790 C0DZ6K 9961315 Ki = 0.34 nM T52790 CNP82Y 9961936 Ki = 0.9 nM T52790 C8CY0E 9961955 Ki = 0.9 nM T52790 C7BG9Z 9981979 IC50 > 5000 nM T52790 CP0I1O 9984184 IC50 = 27 nM T52790 CO7V1Z 9987474 Ki = 13 nM T52790 C3D8BI 10005190 IC50 = 7.7 nM T52790 C73WUR 10010039 Ki = 16 nM T52790 CZ6JW0 10010096 Ki = 11 nM T52790 C1XK9Y 10019102 IC50 > 10000 nM T52790 CWK89Q 10022196 Ki = 3070 nM T52790 CH6DS8 10025594 IC50 > 5000 nM T52790 CEC12Y 10032406 Ki = 7 nM T52790 C71LNR 10032693 Ki = 9 nM T52790 C10WEQ 10041813 IC50 > 5000 nM T52790 CGS3X5 10041814 IC50 > 5000 nM T52790 CEIQ93 10043484 IC50 > 5000 nM T52790 C7AJ2B 10044833 Ki = 2340 nM T52790 CVJ8O1 10045010 IC50 > 5000 nM T52790 C25WVJ 10047566 IC50 > 1000 nM T52790 CRN1L3 10047989 IC50 > 5000 nM T52790 CF6D7J 10055415 IC50 = 65 nM T52790 C7KUO1 10071124 IC50 > 5000 nM T52790 CQN28E 10076881 IC50 = 560 nM T52790 CYOC80 10077113 IC50 = 55 nM T52790 C25LAE 10078301 Ki = 21 nM T52790 COL04Z 10099939 IC50 = 24 nM T52790 C1WVZ0 10102903 Ki = 1597 nM T52790 CGJX24 10121831 Ki = 1.259 nM T52790 CET26N 10122346 Ki = 0.1175 nM T52790 CN8F9Z 10122872 Ki = 31.62 nM T52790 CR1NI5 10145229 Ki = 4.9 nM T52790 C90MXL 10166998 Ki = 0.7943 nM T52790 CTJO63 10167532 Ki = 2.884 nM T52790 CKT51A 10187380 Ki = 2.291 nM T52790 CCBF42 10189341 Ki = 181.97 nM T52790 C0VQ7M 10209751 Ki = 2.399 nM T52790 CC8RL9 10232331 Ki = 1.514 nM T52790 CKEA14 10232332 Ki = 0.2818 nM T52790 C2RYD4 10232566 Ki = 10 nM T52790 C3EC6K 10232846 Ki = 102.33 nM T52790 C8Q9TV 10250427 Ki = 2100 nM T52790 CVQ23E 10258592 IC50 = 177 nM T52790 CD43RZ 10280686 Ki = 4.898 nM T52790 CI87MC 10281234 Ki = 0.631 nM T52790 CP0WB6 10303126 Ki = 5.495 nM T52790 C9XPG3 10303737 Ki = 1.585 nM T52790 CA68DG 10303894 Ki = 0.7586 nM T52790 C9XOF2 10305816 Ki = 3.981 nM T52790 CB8S4N 10318477 IC50 > 5000 nM T52790 CWFB30 10323427 IC50 > 1000 nM T52790 C3C1KJ 10326920 Ki = 0.1585 nM T52790 COJ4A7 10342797 IC50 > 5000 nM T52790 CLN21Y 10349900 IC50 = 17 nM T52790 C1QLH0 10350241 Ki = 31000 nM T52790 CC3UG7 10350454 IC50 = 45 nM T52790 CF5M7J 10350528 IC50 = 46 nM T52790 CWO60K 10350626 IC50 > 10000 nM T52790 CN8PA7 10357986 IC50 > 10000 nM T52790 CZ1J0B 10362340 IC50 > 5000 nM T52790 C92BEU 10364942 IC50 > 5000 nM T52790 CH73CS 10366515 IC50 = 13.4 nM T52790 C6BQR5 10369844 IC50 > 5000 nM T52790 CVQ03A 10370066 Ki = 0.8 nM T52790 C01SWX 10372391 Ki = 3.981 nM T52790 CYSX27 10389807 IC50 > 5000 nM T52790 CK9BP7 10392319 Ki = 4.7 nM T52790 CXG7P5 10393390 IC50 = 389 nM T52790 CKPB41 10394084 IC50 = 6.7 nM T52790 C5V0SZ 10394882 Ki = 2 nM T52790 CV5MR6 10394952 Ki = 21 nM T52790 C1IE7Y 10395141 Ki = 24 nM T52790 C4KZW9 10404051 IC50 > 5000 nM T52790 C49JLI 10410206 IC50 > 5000 nM T52790 CDNR80 10410322 IC50 > 5000 nM T52790 C7EYZ4 10412224 IC50 > 5000 nM T52790 C9A6BX 10417108 Ki = 21 nM T52790 CNX23Q 10429546 IC50 > 5000 nM T52790 CS3P2K 10435115 IC50 = 111 nM T52790 C9JPG8 10435750 IC50 > 5000 nM T52790 C6O1GC 10439730 IC50 = 79 nM T52790 CS57CU 10474902 IC50 > 5000 nM T52790 C31BTI 10477667 IC50 > 5000 nM T52790 CY07LB 10477952 IC50 > 5000 nM T52790 CTFZ13 10477953 IC50 > 5000 nM T52790 CN9WY7 10484667 Ki = 7 nM T52790 CW05ZU 10508281 Ki = 0.1 nM T52790 CD0G5V 10552329 Ki = 33 nM T52790 CW42EP 10554969 Ki = 1258.93 nM T52790 C6F1JR 10576528 Ki = 1258.93 nM T52790 CB1KI8 10578880 Ki = 794.33 nM T52790 CDL4E5 10579116 Ki = 10 nM T52790 CIY19L 10600223 Ki = 22.2 nM T52790 CLJ23U 10603037 Ki = 630.96 nM T52790 C8UEI1 10619783 Ki = 277 nM T52790 CL9UC3 10626894 Ki = 316.23 nM T52790 C5T7OS 10627614 Ki = 7.943 nM T52790 CLOF45 10668461 Ki = 329 nM T52790 CZ1K3M 10691318 Ki = 144 nM T52790 C3JWM0 10696939 Ki = 5.7 nM T52790 C6TEF1 10717843 Ki = 51.6 nM T52790 CY9FS1 10718673 Ki = 6.1 nM T52790 C0AZU9 10722305 Ki = 1.585 nM T52790 C1OBF3 10744541 Ki = 1.5 nM T52790 C7DVG0 10792233 Ki = 1.2 nM T52790 C5XWZ8 10812218 Ki = 172 nM T52790 COH20K 10837820 Ki = 276 nM T52790 CH53JC 10840329 Ki = 1.6 nM T52790 C25BAV 10875000 Ki = 3981.07 nM T52790 CYZ9X4 10875451 Ki = 316.23 nM T52790 C5OQ8E 10876489 Ki = 0.3981 nM T52790 CX65PW 10907460 IC50 = 5180 nM T52790 C4SBO9 10915140 IC50 > 10000 nM T52790 CD8CO5 10929285 IC50 = 0.7943 nM T52790 CEW6Z4 10940813 IC50 = 15.85 nM T52790 CG4A9B 10950925 IC50 = 6.31 nM T52790 CY35LB 10972666 IC50 = 79.43 nM T52790 C39NRJ 10985224 Ki = 398.11 nM T52790 CIT04X 10985363 Ki = 316.23 nM T52790 C1P9YD 10995343 Ki = 1258.93 nM T52790 CJ6EG4 11038500 IC50 = 15.85 nM T52790 CFJG64 11059058 IC50 = 4420 nM T52790 C6XH4P 11181079 Ki = 3.162 nM T52790 C4FWI5 11193639 Ki = 0.1 nM T52790 CC51AU 11193706 Ki = 0.3162 nM T52790 C2QD0L 11203189 Ki = 16 nM T52790 C1O4LI 11205157 Ki = 0.2512 nM T52790 CB7F6K 11205343 Ki = 0.1995 nM T52790 CX8NC7 11216552 Ki = 0.1585 nM T52790 C34XJP 11228042 Ki = 0.1585 nM T52790 CUFQ32 11228450 Ki = 0.1995 nM T52790 CL03PH 11239162 Ki = 0.5012 nM T52790 CAB10S 11239751 Ki = 0.1 nM T52790 CAC71S 11251301 Ki = 5.012 nM T52790 CLSF83 11251435 Ki = 0.3162 nM T52790 C2TC9K 11273015 Ki = 88 nM T52790 C0B1ZR 11274473 Ki = 0.3981 nM T52790 CLS0Z3 11285709 Ki = 0.1995 nM T52790 C47JQX 11285715 Ki = 0.7943 nM T52790 C7NM8R 11285716 Ki = 0.7943 nM T52790 C4G0HZ 11285910 Ki = 3.162 nM T52790 C8SM1W 11296497 Ki = 3.162 nM T52790 C97TFN 11331994 Ki = 0.3981 nM T52790 C9DO3Z 11332007 Ki = 1.995 nM T52790 C0V8EG 11343418 Ki = 1.585 nM T52790 CA0KG1 11366268 Ki = 0.0631 nM T52790 CUR63J 11377052 Ki = 1.995 nM T52790 C5JXZ1 11388737 Ki = 0.1259 nM T52790 CP7KC4 11400251 Ki = 0.3162 nM T52790 CV0O4N 11411718 Ki = 6.31 nM T52790 C6JG9O 11411829 Ki = 0.1585 nM T52790 C07DNR 11421866 Ki = 15.85 nM T52790 C85LYP 11430418 IC50 > 1000 nM T52790 CON8K0 11433617 Ki = 0.05012 nM T52790 CF91HW 11445137 Ki = 0.1 nM T52790 CM9VG7 11468591 Ki = 0.5012 nM T52790 C2L4HE 11479743 Ki = 1.585 nM T52790 C8O9HD 11480157 Ki = 1.259 nM T52790 C93BRP 11491576 Ki = 1.585 nM T52790 C81CAI 11491634 Ki = 0.2512 nM T52790 C7L6JO 11593070 Ki = 0.05754 nM T52790 C1E7TL 11734825 Ki = 457.09 nM T52790 C1KL2C 11764212 Ki = 1 nM T52790 C3BE6W 11764349 Ki = 0.1259 nM T52790 CRJT46 11787612 Ki = 7.943 nM T52790 CX7S5D 11800732 Ki = 4.6 nM T52790 CC9O5K 11801084 Ki = 1258.93 nM T52790 C8K7OQ 11802167 Ki = 19.95 nM T52790 CGHC56 11951302 IC50 = 46000 nM T52790 C8VX6O 14986135 IC50 > 10000 nM T52790 CE01FG 15391369 IC50 = 18 nM T52790 C0OU2J 15485361 IC50 = 3.9 nM T52790 COJ24C 15508105 Ki = 1 nM T52790 CN8XO4 15887536 Ki > 1000 nM T52790 C8N2EM 15887537 Ki = 17 nM T52790 CNF70V 16220269 IC50 = 28000 nM T52790 CA3SL9 18393120 Ki = 20 nM T52790 C3R1FL 18964186 IC50 = 8.9 nM T52790 CCG67R 19610193 Ki = 124 nM T52790 C81JWV 20906619 Ki = 8000 nM T52790 C6ZQC4 21121353 IC50 = 99 nM T52790 CH4PM8 21831101 IC50 = 8.9 nM T52790 CZSA17 22405732 Ki = 33.5 nM T52790 CPL37E 22405734 Ki = 9.9 nM T52790 C9Q2XL 22405735 Ki = 2.1 nM T52790 CXS85F 22405743 Ki = 47 nM T52790 CZF42D 22405753 Ki = 66 nM T52790 CPFZ38 22405758 Ki = 13.1 nM T52790 C7U1ZN 22405761 Ki = 40 nM T52790 CU20GD 22405762 Ki = 9.2 nM T52790 CM67WB 22405764 Ki = 3.7 nM T52790 CHI80E 22901328 Ki = 1770 nM T52790 CXF8Z9 23294208 IC50 = 6.4 nM T52790 C3XN1D 23294214 IC50 = 348 nM T52790 CH68SB 23625179 Ki = 1.95 nM T52790 CA06BR 23625180 Ki = 1.95 nM T52790 C9LGH8 23625320 Ki < 1000 nM T52790 CM36PV 23625321 Ki = 20.89 nM T52790 C45QBV 23625322 Ki = 95.5 nM T52790 C0WAE6 23625323 Ki = 1000 nM T52790 COV6G7 23625324 Ki = 24.55 nM T52790 C5W4OI 23625325 Ki = 0.8511 nM T52790 CGJ8V1 23625326 Ki = 30.2 nM T52790 C8V1WA 23625329 Ki = 0.05248 nM T52790 CQFL68 23625471 Ki = 10.72 nM T52790 CY7F8R 23625473 Ki = 123.03 nM T52790 C7NJC5 23625474 Ki = 91.2 nM T52790 CT9IV8 23625475 Ki = 14.79 nM T52790 CVE7B5 23625476 Ki = 1.38 nM T52790 C28SZX 23625633 Ki = 12.59 nM T52790 CRS41X 23625634 Ki = 4.169 nM T52790 C7FN6J 23625635 Ki = 9.12 nM T52790 CVF4Y8 23625636 Ki = 72.44 nM T52790 CB94KR 23625637 Ki = 3.802 nM T52790 C17VCN 23625783 Ki = 28.18 nM T52790 CTM84P 23625784 Ki = 10.96 nM T52790 C45ZSQ 23625785 Ki = 2.138 nM T52790 CUH60S 23625786 Ki = 25.7 nM T52790 C5K9IB 23625787 Ki = 9.333 nM T52790 CG1D6Y 23625950 Ki = 0.4266 nM T52790 C18LZI 23626108 Ki = 0.8128 nM T52790 C85TXI 23626109 Ki = 3.162 nM T52790 CHFD92 23626110 Ki = 0.1318 nM T52790 C54SCX 23626111 Ki = 2.042 nM T52790 CWY4R5 23626252 Ki = 3.802 nM T52790 CD3KR9 23626253 Ki = 8.511 nM T52790 CAJR25 23626254 Ki = 4.898 nM T52790 CHMR01 23626411 Ki = 4.677 nM T52790 CFU7K4 23626412 Ki = 0.7586 nM T52790 C1HND2 23626413 Ki = 1.072 nM T52790 CN3K1B 23626568 Ki = 0.8913 nM T52790 C6RIV8 23626569 Ki = 1.175 nM T52790 CT12OK 23626743 Ki = 0.2239 nM T52790 CFDH52 23626744 Ki = 0.5495 nM T52790 CU4LO8 23626900 Ki = 0.3715 nM T52790 C92NKR 23627058 Ki = 0.2344 nM T52790 CA97HR 23627059 Ki = 0.06026 nM T52790 CC9H8Z 23627060 Ki = 0.1413 nM T52790 CN54UX 23627061 Ki = 0.09772 nM T52790 CQ4V6M 25071640 Ki = 0.3162 nM T52790 C7NJ1B 25109291 Ki = 3.1 nM T52790 C08BLI 25221995 Ki = 108.6 nM T52790 C3VJ0E 25222441 Ki = 515.3 nM T52790 C2AV1K 44190762 IC50 = 530 nM T52790 CANJ87 44212281 IC50 = 53.2 nM T52790 CJV13F 44212282 IC50 = 16.7 nM T52790 CBFR56 44212283 IC50 = 74 nM T52790 C0WQ8T 44212284 IC50 = 34.2 nM T52790 C1TNM2 44212285 IC50 = 7.02 nM T52790 C46PEF 44215303 Ki = 11 nM T52790 C16DHL 44215305 Ki = 12 nM T52790 CB4CJ8 44215306 Ki = 14 nM T52790 CP37XK 44266422 Ki = 172 nM T52790 C0WK7U 44266459 Ki = 111 nM T52790 CYBO34 44266493 Ki = 82 nM T52790 CQ18SV 44266551 Ki = 316 nM T52790 C5Q9SI 44266599 Ki = 214 nM T52790 CQ04LU 44276673 IC50 = 50 nM T52790 C8YE9F 44276738 IC50 = 204 nM T52790 CPC5E6 44276792 IC50 = 2.5 nM T52790 CM8VY3 44281303 Ki = 17 nM T52790 CT06IA 44281332 Ki = 1 nM T52790 CFZ83O 44281333 Ki = 21 nM T52790 CW6U9X 44281334 Ki = 43 nM T52790 CSEA92 44281342 Ki = 7 nM T52790 C1K3ZC 44281345 Ki = 14 nM T52790 CUYH47 44281358 Ki = 332 nM T52790 CE7JC3 44281359 Ki = 13 nM T52790 CWP8O9 44281391 Ki = 100 nM T52790 C52GFN 44281392 Ki = 118 nM T52790 C13QOA 44281397 Ki = 136 nM T52790 C8B3RD 44281415 Ki = 20 nM T52790 CWC1L5 44281485 Ki = 38 nM T52790 C0TB5X 44281505 Ki = 42 nM T52790 CA1I8S 44281516 Ki = 21 nM T52790 CTVS72 44281538 Ki = 15 nM T52790 CEKC48 44281567 Ki = 9 nM T52790 CQ3W5Y 44281571 Ki = 8 nM T52790 C07XYA 44281572 Ki = 35 nM T52790 CH6UM7 44281587 Ki = 7 nM T52790 CXR0C9 44281633 Ki = 6 nM T52790 C1FK2S 44281649 Ki = 1 nM T52790 CL9IQ2 44281650 Ki = 3 nM T52790 C7S2TC 44281666 Ki = 4 nM T52790 C08YIH 44281672 Ki = 6 nM T52790 C0PKV4 44281680 Ki = 20 nM T52790 C9ZR1S 44281685 Ki = 2 nM T52790 CHV15K 44281713 Ki = 18 nM T52790 C2IC6G 44281722 Ki = 12 nM T52790 C0C8TK 44281723 Ki = 4 nM T52790 CV3U5P 44281726 Ki = 40 nM T52790 CQ92BL 44281743 Ki = 157 nM T52790 C4D1JN 44281744 Ki = 286 nM T52790 C6H5UG 44281753 Ki = 10 nM T52790 CME9G6 44281771 Ki = 28 nM T52790 C37KZY 44281776 Ki = 8 nM T52790 CS4D1T 44281778 Ki = 6 nM T52790 CO6YR1 44281784 Ki = 25 nM T52790 CR62KW 44281785 Ki = 130 nM T52790 C4QZ8K 44281787 Ki = 4 nM T52790 C8AOU7 44281788 Ki = 54 nM T52790 CR2X6V 44281957 Ki = 167 nM T52790 C1S5QC 44281958 Ki = 4 nM T52790 CJ2SU9 44281976 Ki = 2 nM T52790 CZ58US 44281977 Ki = 2 nM T52790 C10-JUN 44282001 Ki = 8 nM T52790 C4O6IF 44282002 Ki = 3 nM T52790 CBE5C7 44282003 Ki = 22 nM T52790 C80LGR 44282004 Ki = 130 nM T52790 CW3OZ0 44300619 Ki = 6.5 nM T52790 C4ZR0P 44300632 Ki = 7.7 nM T52790 C60UKZ 44300668 Ki = 142 nM T52790 CE6L5G 44302393 Ki = 1023.29 nM T52790 CSVJ03 44302394 Ki = 1.479 nM T52790 CY05XI 44302414 Ki = 1.445 nM T52790 CNZQ32 44302496 Ki = 6.607 nM T52790 CXU4N2 44302497 Ki = 1.349 nM T52790 C0N3ZR 44302769 Ki = 24.55 nM T52790 CP56XK 44302816 Ki = 0.1549 nM T52790 CH15KD 44302817 Ki = 87.1 nM T52790 CY5R7N 44305221 IC50 > 1000 nM T52790 C7WI6B 44305248 IC50 = 108 nM T52790 CPI9T3 44305271 IC50 = 500 nM T52790 C1LDB0 44305288 IC50 > 1000 nM T52790 C3V1BM 44305467 IC50 > 1000 nM T52790 C1UBW2 44305511 IC50 = 168 nM T52790 C97DBP 44305544 IC50 = 51 nM T52790 CCHD47 44305557 IC50 = 30 nM T52790 CQY7G9 44305817 Ki = 2400 nM T52790 C04SCG 44305928 Ki = 4200 nM T52790 CHEC65 44308430 EC50 > 50000 nM T52790 CRT79O 44308431 EC50 > 50000 nM T52790 C6ONP4 44308550 EC50 > 50000 nM T52790 CK8W5Q 44308551 EC50 > 50000 nM T52790 CKA2D1 44309945 IC50 = 6.6 nM T52790 CE4X6H 44309946 IC50 = 6.4 nM T52790 CO3D7A 44310102 IC50 = 6.3 nM T52790 CCHX43 44310105 IC50 = 7.1 nM T52790 CMG7B6 44310139 IC50 = 8.4 nM T52790 CRC3A6 44310150 IC50 = 7.3 nM T52790 C8TW9M 44310151 IC50 = 8.1 nM T52790 CX8R3S 44310165 IC50 = 7.7 nM T52790 CKL47H 44310237 IC50 = 6.5 nM T52790 C9MY5S 44310238 IC50 = 7.5 nM T52790 CXR71J 44310262 IC50 = 7.4 nM T52790 C63PEI 44310282 IC50 = 6.7 nM T52790 C2OEW3 44310284 IC50 = 6.3 nM T52790 CN5TI3 44310432 IC50 = 7.2 nM T52790 C7KPM8 44310433 IC50 = 6.8 nM T52790 CS52NG 44310456 IC50 = 6.8 nM T52790 CRFO30 44312000 IC50 = 928 nM T52790 C05TAD 44312026 IC50 > 5000 nM T52790 C1W0GK 44312028 IC50 = 258 nM T52790 CX9PD5 44312056 IC50 = 1400 nM T52790 CIA8X7 44312057 IC50 > 1000 nM T52790 CX2LK5 44312145 IC50 = 211 nM T52790 COT58K 44312169 IC50 = 2100 nM T52790 C1LW7N 44312218 IC50 = 166 nM T52790 C0B2IC 44312219 IC50 = 14 nM T52790 C5V9WG 44312256 IC50 = 4500 nM T52790 C5G3YW 44312257 IC50 = 24 nM T52790 CI7NK6 44312285 IC50 = 4200 nM T52790 CW0C3U 44312324 IC50 = 139 nM T52790 CFK3D2 44312406 Ki = 5010 nM T52790 CK50SI 44312408 Ki > 10000 nM T52790 CM12KY 44312437 Ki > 10000 nM T52790 CPS5B1 44312485 Ki = 4000 nM T52790 CY2H7Q 44312564 Ki = 12600 nM T52790 C2D3KH 44312703 Ki > 10000 nM T52790 CH45RO 44312761 Ki = 12600 nM T52790 CRD1X4 44314154 Ki = 738 nM T52790 CFO10R 44314298 Ki = 259 nM T52790 CA78GB 44314299 Ki = 26 nM T52790 CO84ZW 44314453 Ki > 680 nM T52790 C4O8RX 44314454 Ki = 566 nM T52790 CJTI39 44314476 Ki = 397 nM T52790 CX6Y2B 44314481 Ki = 358 nM T52790 CGY3S5 44314482 Ki = 21 nM T52790 CG9C8F 44314486 Ki = 95 nM T52790 CQ2IB5 44314487 Ki = 48 nM T52790 CYV8U9 44314502 Ki = 30 nM T52790 CQ5W1O 44314503 Ki = 31 nM T52790 CY59OC 44314504 Ki = 33 nM T52790 C43KGB 44314533 Ki = 208 nM T52790 CG7MS4 44314547 Ki = 978 nM T52790 CMX0D9 44314548 Ki = 217 nM T52790 CFK43V 44314577 Ki = 409 nM T52790 C5U8QB 44314578 Ki = 266 nM T52790 CHP4L1 44314597 Ki = 200 nM T52790 C10WAI 44314732 Ki = 477 nM T52790 CF12UM 44314834 Ki = 128 nM T52790 C87BVG 44314865 Ki = 368 nM T52790 CW4L2A 44314866 Ki > 680 nM T52790 CDX9O1 44314867 Ki = 34 nM T52790 C9VZE7 44314868 Ki = 34 nM T52790 CP0L4F 44314871 Ki = 28 nM T52790 CC7VT0 44314872 Ki = 52 nM T52790 CF2SA5 44314873 Ki = 38 nM T52790 CDHG71 44314945 Ki = 382 nM T52790 C4S3BF 44314946 Ki = 170 nM T52790 C3J6QU 44315209 Ki = 2.5 nM T52790 CH30NT 44315210 Ki = 4 nM T52790 C9PT3J 44315231 Ki = 2.8 nM T52790 CM9KT1 44315267 Ki = 2.5 nM T52790 CKT98C 44315297 Ki = 1.2 nM T52790 CAT8U5 44315298 Ki = 1.1 nM T52790 CF50BD 44315299 Ki = 1.2 nM T52790 CF2EQ0 44315369 Ki = 1.5 nM T52790 C70HNK 44315370 Ki = 1.2 nM T52790 C4GLI3 44315390 Ki = 1.7 nM T52790 C1S2MC 44315421 Ki = 3.1 nM T52790 CCW50R 44315422 Ki = 5.2 nM T52790 C46IEH 44315483 Ki = 0.5 nM T52790 C6TRV5 44315572 Ki = 2.6 nM T52790 CS9K4I 44315573 Ki = 4.9 nM T52790 CHX17S 44315576 Ki = 1.8 nM T52790 CDX84T 44315589 Ki = 4.1 nM T52790 C94WGI 44315590 Ki = 3.6 nM T52790 C0UK2L 44315591 Ki = 4.8 nM T52790 C4LP8N 44329148 Ki = 2550 nM T52790 C9N1VT 44329149 Ki = 5580 nM T52790 C5ETU0 44329163 Ki = 17500 nM T52790 C5RQY0 44329339 Ki = 2850 nM T52790 C2HS1R 44329340 Ki = 2240 nM T52790 C8D1PG 44329351 Ki = 6940 nM T52790 CJ8V1U 44329374 Ki = 3440 nM T52790 CY1XC4 44329484 Ki = 3490 nM T52790 C5VXW0 44329517 Ki = 550 nM T52790 CJN80R 44329530 Ki = 4360 nM T52790 CY1DP2 44329531 Ki = 5890 nM T52790 C0TR1M 44331128 Ki = 1.995 nM T52790 CSB4A7 44331207 Ki = 501.19 nM T52790 CEJ6T5 44331223 Ki = 125.89 nM T52790 CDF72P 44332343 Ki = 12.7 nM T52790 C6X0FQ 44332344 Ki = 44.2 nM T52790 CES10Y 44332804 Ki = 156 nM T52790 CTFL83 44332805 Ki > 2000 nM T52790 CK69WY 44332806 Ki > 2000 nM T52790 CXSJ96 44332820 Ki = 1422 nM T52790 CRMZ78 44335318 IC50 = 66 nM T52790 CQRG01 44335319 IC50 = 5.5 nM T52790 C38XWO 44335354 IC50 = 17 nM T52790 C9IB8V 44335360 IC50 = 55 nM T52790 CECZ64 44335372 IC50 = 60 nM T52790 CMF9U8 44335376 IC50 = 26 nM T52790 C3KP7V 44335410 IC50 = 203 nM T52790 CZKP39 44335466 IC50 = 19.5 nM T52790 C62MLD 44336987 Ki > 1000 nM T52790 C5M2EF 44337007 Ki > 1000 nM T52790 C70YEO 44337023 Ki > 1000 nM T52790 C0S1MJ 44337024 Ki > 1000 nM T52790 C2QUC4 44337078 Ki > 1000 nM T52790 COC3Y7 44337079 Ki > 1000 nM T52790 C79RVK 44337080 Ki > 1000 nM T52790 C9KFY3 44337173 Ki = 3 nM T52790 CF0M7V 44337174 Ki = 1.3 nM T52790 CME07I 44337200 Ki > 1000 nM T52790 C1I6ZY 44337201 Ki = 219 nM T52790 C24XSU 44337202 Ki = 8.3 nM T52790 C59BDG 44337207 Ki = 1.1 nM T52790 CG8RD6 44337208 Ki = 1.1 nM T52790 C8A1CW 44337266 Ki = 3.4 nM T52790 C1SUX0 44337270 Ki = 7 nM T52790 CWB0E3 44337288 Ki = 14 nM T52790 CY4XF2 44337289 Ki = 27 nM T52790 C9M2AX 44337308 Ki = 22 nM T52790 CE0XL3 44337313 Ki = 3.4 nM T52790 C1HLR5 44337324 Ki = 28 nM T52790 CNQS47 44337330 Ki = 3.2 nM T52790 CQ6B2X 44337353 Ki = 16 nM T52790 C3TM4J 44337354 Ki = 0.9 nM T52790 CI2TP9 44337355 Ki = 1.3 nM T52790 C8Z4UQ 44337370 Ki = 270 nM T52790 CKT4Z8 44337371 Ki = 14 nM T52790 C7NH1L 44337372 Ki > 1000 nM T52790 CA0QJ4 44337414 Ki = 175 nM T52790 C9EO0J 44337417 Ki > 1000 nM T52790 CU1X6H 44337467 Ki = 300 nM T52790 CA9S5B 44337514 Ki > 1000 nM T52790 CBA09N 44342780 Ki = 3.162 nM T52790 CR5G3L 44342797 Ki = 6.31 nM T52790 CSC35N 44342868 Ki = 12.59 nM T52790 CYTJ53 44342903 Ki = 12.59 nM T52790 C2YFO3 44342904 Ki = 3.981 nM T52790 C93WRP 44343033 Ki = 5.012 nM T52790 CWC30Z 44343083 Ki = 3.162 nM T52790 CTD31C 44343084 Ki = 10 nM T52790 C8EIY1 44343099 Ki = 630.96 nM T52790 C9L2CE 44343142 Ki = 0.3981 nM T52790 CDIK37 44343143 Ki = 7.943 nM T52790 C0IHQ4 44343144 Ki = 1.585 nM T52790 C8Z0LT 44353064 Ki = 2.512 nM T52790 CU3CA8 44353078 Ki = 10 nM T52790 CPK1M0 44363435 Ki = 91 nM T52790 C9JX1F 44363436 Ki = 23 nM T52790 C36NEP 44363442 Ki = 15 nM T52790 C5BGV8 44363756 Ki = 144 nM T52790 CL03EB 44363877 Ki = 146 nM T52790 C4P7HE 44363908 Ki = 4 nM T52790 CLT92R 44363909 Ki = 20 nM T52790 C97AKV 44363912 Ki = 26 nM T52790 C3SJ2T 44363925 Ki = 67 nM T52790 C7W8HN 44363926 Ki = 16 nM T52790 CUS74Z 44363936 Ki = 33 nM T52790 CXOL74 44363948 Ki = 195 nM T52790 C98HSV 44363949 Ki = 23 nM T52790 C5MKE6 44363952 Ki = 11 nM T52790 C4FMW7 44363962 Ki = 28 nM T52790 CO96ZG 44363963 Ki = 27 nM T52790 CN5Z4T 44363978 Ki = 47 nM T52790 C10SMA 44363979 Ki = 53 nM T52790 CM3E7F 44363982 Ki = 39 nM T52790 C8RFG9 44363983 Ki = 16 nM T52790 C0AF2Z 44363984 Ki = 58 nM T52790 C2W8KH 44363990 Ki = 26 nM T52790 CG5H8R 44364001 Ki = 137 nM T52790 C5UK4I 44364002 Ki = 67 nM T52790 CK91IA 44364003 Ki = 59 nM T52790 CY5O2B 44364030 Ki = 39 nM T52790 CK6UC2 44374427 Ki = 1.585 nM T52790 C3OQ6K 44374504 Ki = 7.943 nM T52790 CFGD07 44374543 Ki = 5.012 nM T52790 C26SVP 44374556 Ki = 1.585 nM T52790 C4R7NV 44374557 Ki = 6.31 nM T52790 CW89OL 44374598 Ki = 2.512 nM T52790 CJ10MF 44374622 Ki = 6.31 nM T52790 C5X2HP 44375827 IC50 = 53.36 nM T52790 CE89OF 44375853 IC50 = 7.72 nM T52790 CC7U2B 44379971 IC50 = 25342 nM T52790 C87PLB 44380062 Ki = 1.7 nM T52790 CH7UK2 44380069 Ki = 11.5 nM T52790 CK95JD 44380072 Ki = 0.5 nM T52790 CUP91D 44380079 Ki = 590 nM T52790 C41ZOW 44380081 Ki = 50 nM T52790 CO61AX 44380082 Ki = 8.8 nM T52790 C3Y1FS 44380090 Ki = 3.1 nM T52790 C81BCL 44380091 Ki = 1.5 nM T52790 CAM4W5 44380092 Ki = 23 nM T52790 CKFH38 44380093 Ki = 45 nM T52790 CUD8V6 44380094 Ki = 58 nM T52790 CP1N5F 44380095 Ki = 19 nM T52790 COCK40 44380131 Ki = 3.2 nM T52790 CZ4OK3 44380132 Ki = 3.5 nM T52790 C5W2LY 44380176 IC50 = 14.3 nM T52790 CPC91W 44380206 Ki = 0.8 nM T52790 C3LA4N 44380248 Ki = 5.4 nM T52790 CV0S3A 44380249 Ki = 8.5 nM T52790 CW1RF0 44380277 Ki = 215 nM T52790 CDJ1I5 44380279 Ki = 4.5 nM T52790 C7SU4I 44380289 Ki = 25 nM T52790 CS30MR 44380290 Ki = 17 nM T52790 CAO4I2 44380313 Ki = 236 nM T52790 CGT8P4 44380337 Ki = 4.8 nM T52790 C5YBD1 44380338 Ki = 6.8 nM T52790 C4IE0V 44380396 Ki = 0.7 nM T52790 C93AGV 44380413 Ki = 48 nM T52790 CH0QX3 44380414 Ki = 4.2 nM T52790 CKR3J9 44380415 Ki = 2 nM T52790 C0BO2Q 44380448 Ki = 0.8 nM T52790 C0CN7P 44380457 Ki = 16.7 nM T52790 CI4GR9 44380473 Ki = 394 nM T52790 CJW1X3 44380474 Ki = 350 nM T52790 C2SA3D 44380526 Ki = 1.4 nM T52790 CM7X5R 44380527 Ki = 19 nM T52790 CZ0O9E 44380596 Ki = 42 nM T52790 C7LK2B 44380732 Ki = 14 nM T52790 C2WDA0 44380733 Ki = 50 nM T52790 CHK0I5 44380763 Ki = 107 nM T52790 CO09YI 44380764 Ki = 24 nM T52790 C9Z1VX 44380795 Ki = 198 nM T52790 CNKR49 44384677 IC50 = 42.4 nM T52790 C2JK9W 44384678 IC50 = 96.3 nM T52790 CX0N1K 44384901 IC50 = 11.8 nM T52790 CY43OG 44384902 IC50 = 12 nM T52790 CPRI69 44384986 IC50 = 13.4 nM T52790 C29NBY 44384987 IC50 = 19.1 nM T52790 CD34IL 44385575 IC50 = 55.5 nM T52790 C2CI6G 44386105 IC50 = 548 nM T52790 C0V6SU 44386230 IC50 = 4.04 nM T52790 CR43OB 44386231 IC50 = 6.94 nM T52790 CI83YN 44390434 Ki > 1000 nM T52790 C02SFA 44390446 Ki = 320 nM T52790 C84YPL 44390451 Ki = 310 nM T52790 C7HB2A 44390506 Ki = 500 nM T52790 CYS61B 44390529 Ki = 200 nM T52790 CD26HR 44390532 Ki = 630 nM T52790 C0HR9K 44390533 Ki = 790 nM T52790 CD84XK 44390534 Ki = 5000 nM T52790 C1NP8C 44390535 Ki = 200 nM T52790 CJ2L1E 44390536 Ki > 1000 nM T52790 C9O6DS 44390537 Ki > 200 nM T52790 CU1I8Y 44390539 Ki = 630 nM T52790 CU69PM 44390541 Ki = 120 nM T52790 CO2CJ7 44390546 Ki > 1000 nM T52790 CO36YA 44390550 Ki > 3000 nM T52790 CC71ID 44390552 Ki > 1000 nM T52790 C2YVM0 44390553 Ki = 63 nM T52790 CI3RU0 44390557 Ki > 1000 nM T52790 C14JEM 44390560 Ki = 250 nM T52790 C8LC7H 44390562 Ki > 3000 nM T52790 CMHF80 44390572 Ki > 1000 nM T52790 CK0VL3 44390573 Ki > 100 nM T52790 CACU43 44390574 Ki > 1000 nM T52790 CQ2CS7 44390582 Ki > 3000 nM T52790 C3VIJ9 44390588 Ki = 200 nM T52790 C6ZY8L 44390591 Ki > 310 nM T52790 CC7R0G 44390595 Ki > 1000 nM T52790 C0FWE1 44390600 Ki > 3000 nM T52790 C2BZ3R 44390601 Ki = 130 nM T52790 C0ANU5 44390606 Ki = 200 nM T52790 CEU9G0 44390607 Ki = 50 nM T52790 CRJ32T 44390987 Ki = 2000 nM T52790 CSA8Z6 44390988 Ki > 1000 nM T52790 C1X8SR 44390990 Ki > 3000 nM T52790 CD8R4J 44390991 Ki > 10000 nM T52790 C02IVS 44390992 Ki > 10000 nM T52790 CNB0Z5 44390993 Ki = 7900 nM T52790 CHNA96 44390994 Ki = 2000 nM T52790 CCT3S1 44390995 Ki > 10000 nM T52790 CWES63 44390998 Ki = 200 nM T52790 CN9GF1 44391000 Ki > 1000 nM T52790 CUHZ27 44391001 Ki > 3000 nM T52790 C4C1IO 44391004 Ki > 3000 nM T52790 CD26JS 44391005 Ki = 3000 nM T52790 CG48JP 44391006 Ki = 2000 nM T52790 C08DFQ 44391009 Ki = 6300 nM T52790 C7FP1G 44391011 Ki = 300 nM T52790 C4MC5Y 44391014 Ki > 3000 nM T52790 CQ81TW 44391019 Ki = 10000 nM T52790 CNPT65 44391022 Ki = 5000 nM T52790 C24RKA 44391025 Ki > 1000 nM T52790 CYPV73 44391026 Ki = 3100 nM T52790 C6O7SC 44391030 Ki > 10000 nM T52790 CV4G1U 44391033 Ki = 310 nM T52790 CDR78C 44391034 Ki = 5000 nM T52790 CW26MD 44391036 Ki = 6300 nM T52790 CDTX08 44391037 Ki > 10000 nM T52790 C9RZS4 44391042 Ki > 10000 nM T52790 CPK4G5 44391043 Ki > 1000 nM T52790 CTX97E 44391047 Ki > 10000 nM T52790 C2WKA0 44391051 Ki > 1000 nM T52790 C51LSC 44391061 Ki = 1000 nM T52790 C8ZVM3 44391066 Ki = 790 nM T52790 C54EPN 44391078 Ki = 7900 nM T52790 CH2NF1 44391082 Ki > 1000 nM T52790 CNLS21 44391083 Ki > 3000 nM T52790 CDU0A7 44391084 Ki = 500 nM T52790 CUSZ26 44391089 Ki > 1000 nM T52790 CD0PU8 44391090 Ki > 1000 nM T52790 CK3RO8 44391091 Ki > 3000 nM T52790 C5NL9P 44391095 Ki > 10000 nM T52790 C3GNS2 44391101 Ki > 3000 nM T52790 CHXQ28 44391105 Ki = 100 nM T52790 CU9CZ7 44391106 Ki > 10000 nM T52790 CQ43CH 44391115 Ki > 1000 nM T52790 CJ9WG4 44391116 Ki > 3000 nM T52790 CE9ZS6 44391123 Ki = 3000 nM T52790 CGA56P 44391129 Ki > 1000 nM T52790 CJB14G 44391130 Ki = 1600 nM T52790 C53IJO 44391136 Ki = 1600 nM T52790 CXM26A 44391144 Ki > 1000 nM T52790 C0AP6L 44391145 Ki = 2000 nM T52790 CKB2M9 44391153 Ki = 600 nM T52790 CT03BE 44392318 Ki = 9500 nM T52790 C6MRW3 44392347 IC50 = 7.943 nM T52790 C9AG0M 44392351 IC50 = 1.259 nM T52790 C2TM3S 44392392 IC50 = 3.162 nM T52790 CLO40U 44392439 IC50 = 1.259 nM T52790 C3X2LP 44392444 IC50 = 10 nM T52790 C8F0YB 44392445 IC50 = 2.512 nM T52790 CDB14V 44392491 IC50 = 1 nM T52790 CY4X5F 44392497 Ki = 10000 nM T52790 CI6O9K 44402934 IC50 = 49 nM T52790 CX6V9Q 44404006 IC50 = 2.25 nM T52790 CGZ2J9 44411637 IC50 = 550 nM T52790 CE45QC 44411742 IC50 = 1000 nM T52790 CS0IE2 44421488 Ki = 0.0631 nM T52790 CL3OX6 44421489 Ki = 0.05012 nM T52790 C3RD0X 44421490 Ki = 0.1995 nM T52790 CO7AX5 44421491 Ki = 1.585 nM T52790 CZ7AE5 44421492 Ki = 25.12 nM T52790 C2TSZ9 44421493 Ki = 0.631 nM T52790 C1UH6T 44421494 Ki = 0.5012 nM T52790 CN10HJ 44421495 Ki = 3.981 nM T52790 C9MIJ5 44434158 Ki = 70.79 nM T52790 C7XD6K 44434159 Ki = 10000 nM T52790 CS35EM 44434160 Ki = 316.23 nM T52790 CX24CV 44434161 Ki = 50.12 nM T52790 C1RQ6E 44434162 Ki = 316.23 nM T52790 CG19CO 44434163 Ki = 316.23 nM T52790 CS2JL7 44434164 Ki = 39.81 nM T52790 C8BQL5 44434166 Ki = 398.11 nM T52790 CGZL15 44434168 Ki = 12.59 nM T52790 C5IC2K 44434169 Ki = 125.89 nM T52790 C0XTR4 44434170 Ki = 50.12 nM T52790 CCD86T 44434171 Ki = 19.95 nM T52790 C05LRK 44434174 Ki < 1000 nM T52790 C7LT5B 44434175 Ki = 100 nM T52790 CMP41Z 44434176 Ki < 10000 nM T52790 CJR0B1 44434177 Ki = 251.19 nM T52790 CFSH86 44434178 Ki = 100 nM T52790 C94XDI 44434179 Ki = 100 nM T52790 C3J0FB 44434180 Ki = 6.31 nM T52790 CG15WE 44434181 Ki = 125.89 nM T52790 C5TAY7 44434182 Ki = 100 nM T52790 CL7CX1 44434183 Ki = 63.1 nM T52790 CX14ZR 44434184 Ki = 19.95 nM T52790 CD6J3M 44434185 Ki = 3.981 nM T52790 CZ83PS 44434186 Ki = 31.62 nM T52790 CAP0J9 44434187 Ki = 100 nM T52790 CG9O2B 44434188 Ki = 50.12 nM T52790 C5BAY7 44434189 Ki = 25.12 nM T52790 CL8Z5R 44434190 Ki = 7.943 nM T52790 C8T4HV 44434191 Ki = 0.3981 nM T52790 CGL98K 44434192 Ki = 100 nM T52790 CJB9Y1 44434193 Ki = 3.981 nM T52790 CKG4Y6 44434194 Ki = 1.995 nM T52790 CF8B9V 44434195 Ki = 1.585 nM T52790 CYL6U0 44434196 Ki = 1.259 nM T52790 C8QES2 44434197 Ki = 1.995 nM T52790 C7BWO8 44434198 Ki = 1 nM T52790 C20YMJ 44434202 Ki = 1.585 nM T52790 C7PO6W 44434203 Ki = 1.259 nM T52790 CNKM72 44434204 Ki = 1.995 nM T52790 CVFX98 44434205 Ki = 2.512 nM T52790 C1H7YR 44444681 IC50 = 1730 nM T52790 CPMZ84 44458598 IC50 > 5000 nM T52790 CX0TU1 44458983 IC50 > 5000 nM T52790 C0GUN2 44459032 IC50 > 5000 nM T52790 C4DL5C 44469677 IC50 > 10000 nM T52790 CG1QT9 44550460 Ki = 952.6 nM T52790 CHI2Y7 44577884 Ki = 25.12 nM T52790 C9DCV4 44577885 Ki = 19.95 nM T52790 C12SJR 44577886 Ki = 5.012 nM T52790 C5SI6D 44577887 Ki = 3.981 nM T52790 C0AF9X 44577888 Ki = 3.981 nM T52790 CJ5MI0 44577889 Ki = 10 nM T52790 C52QEU 44577890 Ki = 7.943 nM T52790 CZQ7D0 44577891 Ki = 12.59 nM T52790 C8PE2T 44577892 Ki = 3.162 nM T52790 C2J4WS 44577893 Ki = 0.7943 nM T52790 C0RNV2 44577894 Ki = 10 nM T52790 CTDN82 44577895 Ki = 5.012 nM T52790 CJ2DX5 44577896 Ki = 25.12 nM T52790 CV1OH0 44577897 Ki = 3.981 nM T52790 CUBZ68 44577898 Ki = 1 nM T52790 CJ9D0M 44577899 Ki = 1.995 nM T52790 CC1E3Q 44577900 Ki = 1 nM T52790 CW2BQ6 44577901 Ki = 1.259 nM T52790 C4S9JF 44577902 Ki = 1.259 nM T52790 C2G7PI 44577903 Ki = 0.7943 nM T52790 CIQ01W 44577904 Ki = 1.995 nM T52790 CH53JX 44577905 Ki = 1.585 nM T52790 CFNX45 44577906 Ki = 1 nM T52790 C65MAR 44577907 Ki = 0.5012 nM T52790 CX7P4A 44577908 Ki = 1 nM T52790 C2VF9P 44577909 Ki > 100 nM T52790 CH6Y8N 44577910 Ki = 15.85 nM T52790 C3IY6C 44577911 Ki = 0.3162 nM T52790 C0JR4P 46236387 Ki = 0.2512 nM T52790 CO7BE5 46236392 Ki = 1 nM T52790 CZI43T 46236394 Ki = 0.3162 nM T52790 C36OWY 46236396 Ki = 0.3162 nM T52790 CT1E7P 46236510 Ki = 0.3981 nM T52790 CO7J2F 46236512 Ki = 0.3981 nM T52790 CW56DU 46236514 Ki = 0.5012 nM T52790 CAYQ64 46236516 Ki = 0.3162 nM T52790 CY6D0I 46236647 Ki = 0.5012 nM T52790 CQE3Z5 46236649 Ki = 1.259 nM T52790 CAMI94 46236655 Ki = 0.5012 nM T52790 C6T9QX 46236794 Ki = 1.995 nM T52790 CE23LJ 46236796 Ki = 0.7943 nM T52790 CH3O5T 46236798 Ki = 0.5012 nM T52790 CBC95E 46236800 Ki = 15.85 nM T52790 CDSB90 46236920 Ki = 0.1259 nM T52790 CIU49M 46237033 Ki = 0.07943 nM T52790 C0Q8GD 46237037 Ki = 0.631 nM T52790 CGO89S 46237038 Ki = 0.2512 nM T52790 CA8YC3 46237168 Ki = 0.631 nM T52790 C2BF3Y 46237169 Ki = 0.7943 nM T52790 CLHX34 46237170 Ki = 0.1259 nM T52790 CMG85O 46237171 Ki = 0.1585 nM T52790 CJI4Q0 46237296 Ki = 1 nM T52790 CM38CH 46237299 Ki = 0.3162 nM T52790 C1TI9K 46237300 Ki = 0.2512 nM T52790 CDJ9H1 46237301 Ki = 0.1585 nM T52790 C4Y0BX 46237302 Ki = 0.1585 nM T52790 CGWN92 46237442 Ki = 1.995 nM T52790 CHLB52 46237445 Ki = 0.1585 nM T52790 C8TQ5C 46237575 Ki = 1.995 nM T52790 C95RWS 46237698 Ki = 0.631 nM T52790 C79QMZ 46237825 Ki = 0.631 nM T52790 CR0W6U 46237957 Ki = 0.5012 nM T52790 C0KMH6 46237960 Ki = 0.3162 nM T52790 CG8S5J 46238091 Ki = 0.631 nM T52790 C7XKM8 46238093 Ki = 0.2512 nM T52790 C30KGU 46238229 Ki = 0.631 nM T52790 C0G4TW 46238232 Ki = 0.3981 nM T52790 CAW09X 46889639 Ki = 1.995 nM T52790 CWV6A0 46889640 Ki = 0.3162 nM T52790 CL0N3Q 46889641 Ki = 0.07943 nM T52790 C8UP2L 46889663 Ki = 0.631 nM T52790 CSU0E2 46889664 Ki = 0.7943 nM T52790 C93GXR 51003494 Ki = 75 nM T52790 CD2YU8 51351496 Ki = 10000 nM T52790 C2UG4W 51351504 Ki = 13000 nM T52790 CK5BW0 52918297 Ki = 2.042 nM T52790 CMG39F 52918298 Ki = 26.92 nM T52790 C9A7NX 52918299 Ki = 44.67 nM T52790 CBM03W 53317584 Ki = 8.318 nM T52790 CBKP15 53318867 Ki = 0.2344 nM T52790 CQB9C6 53322827 Ki = 3.236 nM T52790 CU70SC 53324157 Ki = 0.3236 nM T52790 CWQ64K 53325456 Ki = 4.571 nM T52790 CJRA97 53326714 Ki = 3.981 nM T52790 CK1C9O 53472113 Ki = 794.33 nM T52790 CM2NZ1 54537190 Ki = 0.84 nM T52790 CEFT05 54583959 Ki = 19000 nM T52790 C7CDR5 57391132 Ki = 398000 nM T52790 C02MLR 57391133 Ki = 100000 nM T52790 CH3BG0 57394644 Ki > 3000000 nM T52790 C9AIN2 57396389 Ki = 250000 nM T52790 CLN40O 71449072 IC50 = 43 nM T52790 CCE72K 71449092 Ki = 27000 nM T52790 C8K4ZQ 71449111 Ki = 0.05012 nM T52790 C2CV5X 71449112 Ki = 3.981 nM T52790 CU65NS 71449143 IC50 = 70 nM T52790 C4D8GV 71450855 IC50 = 27 nM T52790 C6WEU0 71450941 IC50 = 28 nM T52790 C3DW2Y 71450949 IC50 = 577 nM T52790 C2MA1K 71452663 IC50 = 123 nM T52790 CBX3C5 71452678 IC50 = 181 nM T52790 CE05UB 71452717 Ki = 0.1259 nM T52790 C8RCG9 71456198 IC50 = 162 nM T52790 C2YIK9 71457960 Ki > 2000 nM T52790 C18VLH 71458000 IC50 = 46 nM T52790 C7PEX9 71458042 Ki = 0.631 nM T52790 C6H2WN 71458099 IC50 = 300 nM T52790 C2C0MK 71458131 IC50 = 120 nM T52790 CST7B2 71461644 Ki = 10 nM T52790 CUXL38 71461646 Ki = 5 nM T52790 C60PAY 71461711 Ki = 2.7 nM T52790 CN8CM1 71533722 Ki = 12589.25 nM T52790 CV47CJ 71549769 Ki = 12589.25 nM T52790 CWH6T3 72548703 IC50 = 1.2 nM T52790 CEA84Y 73347011 Ki = 73000 nM T52790 C8A1DU 73350088 Ki > 100000 nM T52790 CQ0J3N 73350089 Ki = 2400 nM T52790 CU7Q1N 73351501 IC50 = 850 nM T52790 C4SKT9 73351579 Ki = 3800 nM T52790 C5BPU2 73352970 IC50 = 730 nM T52790 CO25EH 73353047 Ki = 33000 nM T52790 C7PK2H 73353048 Ki > 100000 nM T52790 CN8D6S 73354569 Ki > 100000 nM T52790 C9FVI0 73354570 Ki = 1600 nM T52790 CD5W6K 90417914 Ki = 10000 nM T52790 C0AJ4Q 90663622 Ki = 12.59 nM T52790 CH08TW 90663623 Ki = 398.11 nM T52790 CJ06SU 91535935 IC50 = 100 nM T52790 C9ZUP4 91809194 IC50 > 10000 nM T52790 CNS4V9 102531123 IC50 > 10000 nM T52790 CXL57K 102531124 IC50 > 10000 nM T52790 CY8R0C 102531125 IC50 > 10000 nM T52790 C0OSW4 102531127 IC50 > 10000 nM T52790 CWI56P 118724118 Ki = 1.349 nM T52790 C5KW0B 118724119 Ki = 1.479 nM T52790 C3U5IE 118724120 Ki = 1.585 nM T52790 C6GQ2Y 118724121 Ki = 8.318 nM T52790 C4VZK9 118724122 Ki = 5.888 nM T52790 CH1EI7 118724123 Ki = 1949.84 nM T52790 CNGQ19 122179477 IC50 = 4280 nM T52790 C76XAE 125111645 IC50 > 10000 nM T52790 C27PAJ 127032997 IC50 = 3.5 nM T52790 CO4N2F 127034660 IC50 > 10000 nM T52790 CNQ2Y4 127034696 IC50 > 10000 nM T52790 CRAC83 127034748 IC50 > 10000 nM T52790 CV9Z2G 127034749 IC50 > 10000 nM T52790 CJ7T9U 127034767 IC50 > 10000 nM T52790 CE9Z2Y 127034768 IC50 > 10000 nM T52790 C7CYF5 127034769 IC50 > 10000 nM T52790 CNX2F4 127034928 IC50 > 10000 nM T52790 CATQ52 127034940 IC50 > 10000 nM T52790 CL6OW2 127035038 IC50 > 10000 nM T52790 C1AG9R 127035039 IC50 > 10000 nM T52790 C8WXA7 127035040 IC50 > 10000 nM T52790 CE62OX 127035105 IC50 > 10000 nM T52790 CHAS82 127035106 IC50 > 10000 nM T52790 CJR2D5 127035222 IC50 > 10000 nM T52790 C52ALH 127035367 IC50 > 10000 nM T52790 C2S8IW 127035368 IC50 > 10000 nM T52790 CUV12X 127035512 IC50 > 10000 nM T52790 C9PDL3 127035576 IC50 > 10000 nM T52790 CS78HG 127035706 IC50 > 10000 nM T52790 C2PL6V 127036728 IC50 > 10000 nM T52790 C1JKC0 135430775 IC50 > 1000 nM T52790 C1Y3IB 135449286 IC50 = 7 nM T52790 CX2QG6 137633652 Ki = 2 nM T52790 CTD69B 137647980 IC50 = 1300 nM T52790 C6ZU0A 145949555 IC50 > 20000 nM T52790 CE3D8P 145951877 IC50 > 20000 nM T52790 CI9BO4 145952624 IC50 = 3220 nM T52790 CL42TO 145953024 IC50 = 1790 nM T52790 CR2QH0 145957924 IC50 = 4610 nM T52790 CP25CA 145958767 IC50 = 5510 nM T52790 C01GKQ 145971455 IC50 > 20000 nM T52790 C72EFN 155551678 Ki = 0.4 nM T52790 C4AG0H 155558726 Ki = 1600 nM T52790 CR12DI 155565189 Ki = 140 nM T52790 D00HAJ 73347136 IC50 = 710 nM T52790 D00HUY 10473960 IC50 > 5000 nM T52790 D01NPA 5311311 Ki = 0.71 nM T52790 D05ZUX 44207909 Ki >= 1000 nM T52790 D07NNN 5311312 Ki = 15.85 nM T52790 D0A1DE 10917690 IC50 = 3388 nM T52790 D0C7LY 11496610 Ki = 330 nM T52790 D0J8SU 36511 Ki = 102 nM T52790 D0S9CI 11989776 IC50 = 50 nM T52790 D0T2RY 9948320 Ki >= 1000 nM T52790 D0W3XD 16049828 IC50 > 1000 nM T52790 D0Z6TG 9852253 Ki = 0.6 nM T11288 D0BP9C 193962 IC50 = 8500 nM T11288 D0K8KX 5280343 Ki = 2400 nM T11288 D0O3OS 104850 Ki = 1400 nM T11288 D0R0FE 2520 EC50 = 1925 nM T11288 D0R1RS 3715 IC50 = 12000 nM T11288 D0R3JB 4212 IC50 = 27.5 nM T11288 D0Z3DY 2333 Ki = 190 nM T11288 D02HTD 25167947 IC50 = 14900 nM T11288 D02QWY 24785538 IC50 = 36300 nM T11288 D0G7UX 5284373 EC50 = 1700 nM T11288 D0O2EF 56946615 IC50 > 100000 nM T11288 D0V7UQ 56946834 IC50 = 2500 nM T11288 D02VJY 3037617 IC50 = 5180 nM T11288 D07GTB 16760063 IC50 = 7570 nM T11288 C52MFS 1756 EC50 = 42000 nM T11288 C8C1JP 72343 IC50 = 38320 nM T11288 C5ZCH7 97332 IC50 = 26350 nM T11288 CL97OF 97548 IC50 = 9860 nM T11288 CA3NK8 193841 EC50 = 5100 nM T11288 CR67FB 243037 EC50 > 100000 nM T11288 CABJ72 276138 IC50 = 1760 nM T11288 CM70RQ 285815 IC50 = 16000 nM T11288 CN8ZL4 298546 EC50 = 45000 nM T11288 C7HME8 439246 Ki = 2400 nM T11288 COI2C9 560674 EC50 = 98000 nM T11288 CTF2J0 687260 EC50 > 100000 nM T11288 CH6MV7 715632 IC50 = 8770 nM T11288 C64RUF 877998 IC50 = 15900 nM T11288 CXR0P5 917533 IC50 = 8800 nM T11288 C7D1QN 921567 EC50 > 100000 nM T11288 CK8TP4 1019287 IC50 > 100000 nM T11288 CL27VW 1069464 IC50 = 3900 nM T11288 CXQ4P8 1183964 IC50 = 8130 nM T11288 CQT4J5 2094802 IC50 > 100000 nM T11288 C1A0FV 2298706 EC50 = 9800 nM T11288 CW6SA0 2787558 IC50 > 100000 nM T11288 C8PN0C 5280682 IC50 = 50000 nM T11288 CNI9X4 5281888 Ki = 600 nM T11288 CPHR19 5325373 EC50 > 100000 nM T11288 CJMT13 5325385 EC50 > 100000 nM T11288 C8VZ9T 5325386 EC50 > 100000 nM T11288 C81ZSW 5325387 EC50 = 85000 nM T11288 CTO51S 5352005 IC50 = 50000 nM T11288 CB2U6E 5467200 IC50 = 1100 nM T11288 C0EM5S 6509849 IC50 = 2800 nM T11288 C32UFI 9828452 IC50 = 61 nM T11288 C82UNW 9828532 IC50 = 1800 nM T11288 CI78PM 9848185 IC50 = 1050 nM T11288 C30DJS 9873998 IC50 = 800 nM T11288 CK5L6J 9904482 EC50 = 64000 nM T11288 CHI5S9 9975676 IC50 = 2900 nM T11288 CEG64W 9976758 EC50 = 2800 nM T11288 CDTB42 9979854 IC50 >= 250 nM T11288 CL5ZS9 9980860 IC50 = 650 nM T11288 C2B0CY 10004696 IC50 >= 250 nM T11288 CQI0Z7 10029563 IC50 = 76 nM T11288 C0HN4T 10031184 IC50 = 118 nM T11288 CG3RA9 10046544 IC50 = 1850 nM T11288 C5IQ2D 10047863 IC50 < 250 nM T11288 CK4A1L 10048669 IC50 = 1020 nM T11288 C2ZUK8 10051663 IC50 < 250 nM T11288 CC6U1G 10071405 IC50 >= 250 nM T11288 CSY05M 10072430 IC50 = 38 nM T11288 CO0QB1 10092403 IC50 = 7350 nM T11288 CWJ7R4 10094280 IC50 >= 250 nM T11288 CE6X4R 10221081 EC50 = 49100 nM T11288 C96LOC 10251349 IC50 > 50000 nM T11288 CQT7H4 10320818 IC50 = 65 nM T11288 C3I4DW 10322116 IC50 = 715 nM T11288 CY73KI 10322450 EC50 = 1800 nM T11288 CW6D4S 10333981 IC50 = 10800 nM T11288 CK9SQ7 10344755 IC50 = 533 nM T11288 CXG67L 10345205 IC50 = 500 nM T11288 C7Z4DU 10346312 IC50 >= 250 nM T11288 C7Z8IW 10379829 IC50 = 2870 nM T11288 CAO02N 10383921 IC50 = 789 nM T11288 CQU08N 10388318 IC50 >= 250 nM T11288 C36PIN 10407830 IC50 = 197 nM T11288 C1DYS4 10432300 IC50 = 920 nM T11288 CG40WP 10454772 IC50 = 910 nM T11288 CW4BK0 10455921 IC50 = 138 nM T11288 CE7IT1 10459316 IC50 >= 250 nM T11288 CCS90U 10472817 IC50 = 714 nM T11288 C78HZG 10495050 IC50 = 932 nM T11288 CE1U9A 10517005 EC50 > 100000 nM T11288 CCG5H3 10518339 IC50 = 14500 nM T11288 C8HWT1 10543161 IC50 = 2710 nM T11288 CD2EQ3 10585756 IC50 = 43100 nM T11288 CHE31J 10591449 IC50 > 100000 nM T11288 C58EFZ 10616146 IC50 = 4190 nM T11288 CH1V7U 10708375 IC50 = 20400 nM T11288 C7ANU6 10709061 IC50 = 8290 nM T11288 CH72SE 10709378 IC50 = 18300 nM T11288 CSK86O 10756523 IC50 = 2560 nM T11288 C01KTG 10758537 IC50 = 5970 nM T11288 CQF21J 10776189 IC50 = 26400 nM T11288 CI1RC8 10830017 IC50 = 4060 nM T11288 COHV95 10848828 IC50 = 4460 nM T11288 C53AIX 10850200 IC50 = 43400 nM T11288 C2BXZ1 11156535 IC50 >= 250 nM T11288 CKJ32I 11164648 IC50 = 6350 nM T11288 C5E8LY 11168500 IC50 = 20 nM T11288 C84PJK 11177283 IC50 = 94 nM T11288 C8HF7R 11177641 IC50 = 399 nM T11288 CYQ98P 11179994 IC50 = 138 nM T11288 CN3B9L 11186582 IC50 = 9000 nM T11288 CTBH70 11189272 IC50 = 2800 nM T11288 C8CWV4 11200621 IC50 = 632 nM T11288 C6XUE4 11201011 IC50 = 33 nM T11288 CLT87I 11212921 IC50 = 41 nM T11288 CFD6R7 11213871 IC50 = 48 nM T11288 CD8VO1 11214464 IC50 = 15 nM T11288 C63QRZ 11226516 IC50 = 17 nM T11288 C7PTZ8 11246811 IC50 >= 250 nM T11288 C79PBA 11247947 IC50 = 59 nM T11288 C86MWN 11249529 IC50 = 13.7 nM T11288 COJD26 11258566 IC50 = 2300 nM T11288 CEN76W 11261262 IC50 = 40.9 nM T11288 CI1M9O 11270541 IC50 = 28 nM T11288 CP13GR 11270563 IC50 = 59 nM T11288 C8NL3A 11281999 IC50 = 3440 nM T11288 C4I2ZV 11293873 IC50 = 2710 nM T11288 CY79US 11293906 IC50 = 110 nM T11288 CFX64S 11293909 IC50 = 166 nM T11288 CH7E1O 11293927 IC50 = 147 nM T11288 C1YH6T 11295806 IC50 = 97 nM T11288 CJYA49 11304370 IC50 = 24 nM T11288 CXKY42 11305058 IC50 = 45 nM T11288 CD9SN8 11316308 IC50 = 167 nM T11288 CE4HY2 11318194 IC50 = 88 nM T11288 CL8ZT6 11327691 IC50 = 3150 nM T11288 CY8G5H 11337594 IC50 >= 250 nM T11288 C78BGT 11339085 IC50 = 169 nM T11288 C65ZTX 11350733 IC50 = 820 nM T11288 C8P1QC 11351150 IC50 >= 250 nM T11288 CYZ51K 11359019 IC50 = 8370 nM T11288 C61ARN 11362459 IC50 = 1415 nM T11288 C31PLX 11376266 IC50 = 29 nM T11288 CZ9W0I 11385818 IC50 = 78 nM T11288 C8S3OV 11396606 IC50 = 87 nM T11288 C0G4AF 11408751 IC50 = 120 nM T11288 C13MRQ 11418752 IC50 = 955 nM T11288 CUO79V 11419244 IC50 = 63 nM T11288 C49LBJ 11432257 IC50 = 620 nM T11288 CTK09U 11443156 IC50 = 13 nM T11288 CLB97A 11443942 IC50 = 26.5 nM T11288 CM2J9W 11444700 IC50 < 250 nM T11288 CSK8F9 11453657 IC50 = 190 nM T11288 C19WQH 11454150 IC50 >= 250 nM T11288 CTQS76 11454703 IC50 = 10 nM T11288 C59DBU 11454819 IC50 < 250 nM T11288 CYCB17 11455462 IC50 = 107 nM T11288 C6W0MU 11477947 IC50 = 122 nM T11288 CH0T1B 11488138 IC50 = 27 nM T11288 CJXT34 11751643 IC50 = 67 nM T11288 CXWU95 11752839 IC50 < 250 nM T11288 C9X6DU 11774980 IC50 = 51 nM T11288 CLR59J 11775287 IC50 = 62 nM T11288 C2C3WI 11957988 IC50 > 20000 nM T11288 CG1CU7 12219475 EC50 > 100000 nM T11288 CS4D6C 12405466 EC50 = 15100 nM T11288 C4D7RX 12613559 EC50 = 26500 nM T11288 C6UJA5 13144102 EC50 > 100000 nM T11288 CT0DU8 13633111 IC50 = 20400 nM T11288 CO9ES2 13633119 IC50 = 1210 nM T11288 CJ9Z4M 15290116 EC50 = 72000 nM T11288 CLD92G 15999199 IC50 = 40600 nM T11288 C0A3IV 16092354 IC50 = 3730 nM T11288 CMVW98 16618023 EC50 = 728 nM T11288 CX06NR 17412108 IC50 = 39300 nM T11288 CB7T2K 20963109 IC50 = 7720 nM T11288 CFI13S 22310708 IC50 = 7820 nM T11288 CK4UG1 23323164 IC50 > 100000 nM T11288 C3ESV6 24178402 EC50 = 2800 nM T11288 C60EJI 25113688 EC50 = 9300 nM T11288 C6O2ZR 25225119 EC50 = 2700 nM T11288 C3J8PO 39176758 IC50 > 100000 nM T11288 CG7UZ6 44220872 IC50 = 12300 nM T11288 C8C9MJ 44220873 IC50 = 42600 nM T11288 CSLJ20 44220874 IC50 = 5380 nM T11288 CPIM70 44220875 IC50 = 21600 nM T11288 C01FMP 44220876 IC50 = 16200 nM T11288 C04ZKP 44220877 IC50 = 18300 nM T11288 CY9AW0 44221092 IC50 = 11600 nM T11288 C0X8OT 44221093 IC50 = 4510 nM T11288 C12MDG 44221095 IC50 = 14300 nM T11288 C3MNS1 44221096 IC50 = 27500 nM T11288 C2VWE1 44221097 IC50 = 1230 nM T11288 C9BNA1 44248179 EC50 = 73 nM T11288 CKA6N2 44276937 IC50 = 122 nM T11288 CTOA75 44368818 IC50 = 2020 nM T11288 CPLV23 44368900 IC50 > 10000 nM T11288 C26MFU 44368902 IC50 = 7600 nM T11288 CHO6P8 44368923 IC50 = 400 nM T11288 COWL28 44369026 IC50 = 1330 nM T11288 CDLX46 44369027 IC50 = 1560 nM T11288 C9VXD2 44369028 IC50 = 3840 nM T11288 CT0SK1 44369032 IC50 = 36000 nM T11288 CCD76W 44369044 IC50 = 37000 nM T11288 C1V6QO 44369052 IC50 = 900 nM T11288 CY08UQ 44369067 IC50 = 1000 nM T11288 C0FXA2 44369069 IC50 = 18570 nM T11288 C82JKC 44369082 IC50 = 1500 nM T11288 C0Z4TJ 44369087 IC50 = 15100 nM T11288 CZD46M 44369091 IC50 = 6350 nM T11288 CLIY42 44369110 IC50 = 1000 nM T11288 CTE65O 44369198 IC50 = 7200 nM T11288 C1J6DA 44369228 IC50 = 4500 nM T11288 CKPW47 44369229 IC50 = 3200 nM T11288 CA0PF4 44369232 IC50 > 100000 nM T11288 CU9H3K 44369247 IC50 = 39000 nM T11288 C05EUO 44369260 IC50 = 3330 nM T11288 CGU9Z8 44369264 IC50 = 2910 nM T11288 C5JLT0 44369265 IC50 = 2800 nM T11288 CE32OY 44369278 IC50 = 10000 nM T11288 C40XPZ 44404554 IC50 >= 250 nM T11288 CU97QG 44404555 IC50 < 250 nM T11288 CHX57V 44404558 IC50 < 250 nM T11288 C89BQU 44405535 EC50 = 420 nM T11288 CLV54W 44405572 EC50 = 250 nM T11288 C8A7CS 44405716 EC50 = 640 nM T11288 CM8O3W 44451264 EC50 > 100000 nM T11288 C45VCM 44451857 EC50 = 21000 nM T11288 CG61YX 44542293 EC50 > 100000 nM T11288 CI9VZ6 44542743 EC50 > 100000 nM T11288 C80EVI 44723582 EC50 > 100000 nM T11288 C43FNG 45266957 IC50 = 4180 nM T11288 C8C4ZS 45267881 IC50 = 22800 nM T11288 C8IYJ2 45268774 IC50 = 198000 nM T11288 CUE5Y2 45269621 IC50 = 29100 nM T11288 CJG13Y 45272176 IC50 = 24000 nM T11288 CAPW24 45272182 IC50 = 20700 nM T11288 COA30H 46227751 IC50 > 20000 nM T11288 CLWR13 46227752 IC50 > 20000 nM T11288 CX2EU1 46843551 EC50 = 13000 nM T11288 CON7Q5 46888534 EC50 = 46000 nM T11288 C53NLD 46888535 EC50 = 7610 nM T11288 CWO79T 46899560 EC50 = 12000 nM T11288 CUFI19 46899561 EC50 = 8700 nM T11288 C43WPR 46899562 EC50 = 8000 nM T11288 C2QX3P 46899563 EC50 = 63000 nM T11288 CBWT20 46899565 EC50 = 13600 nM T11288 CHR49C 46899724 EC50 > 100000 nM T11288 CZXN91 46899725 EC50 = 85800 nM T11288 C7ZS6E 46899726 EC50 = 29500 nM T11288 C1H9ML 56764960 IC50 = 22700 nM T11288 C2WYN9 56945196 IC50 > 100000 nM T11288 C7RW8P 56945197 IC50 = 11200 nM T11288 C7LDX6 56945198 IC50 > 100000 nM T11288 C2N8DS 56945199 IC50 > 100000 nM T11288 CN2WF6 56945201 IC50 > 100000 nM T11288 CB7W4E 56945202 IC50 > 100000 nM T11288 CT4BW6 56945299 IC50 > 100000 nM T11288 CTEJ21 56945300 IC50 = 45800 nM T11288 CU2HC7 56945301 IC50 = 40600 nM T11288 CUK5Q9 56945302 IC50 = 38800 nM T11288 C36HTV 56945303 IC50 = 46600 nM T11288 C7X2EU 56945304 IC50 = 44500 nM T11288 C4VNX9 56945305 IC50 = 16300 nM T11288 C1JCB9 56945418 IC50 = 44000 nM T11288 C6UD7F 56945419 IC50 = 32200 nM T11288 C98UJH 56945420 IC50 = 8000 nM T11288 C51PRX 56945421 IC50 = 22000 nM T11288 CES25H 56945422 IC50 = 9500 nM T11288 C2QB4L 56945423 IC50 = 7700 nM T11288 CA6UX7 56945524 IC50 = 74500 nM T11288 C4AVC1 56945525 IC50 = 40600 nM T11288 CC25LY 56945526 IC50 = 75800 nM T11288 C8KLW6 56945527 IC50 = 37900 nM T11288 C6ZSA3 56945528 IC50 = 30000 nM T11288 C2IAL8 56945529 IC50 = 28000 nM T11288 CP6G0O 56945530 IC50 > 100000 nM T11288 C27RQI 56946614 IC50 > 100000 nM T11288 CK1ZU5 56946616 IC50 = 23600 nM T11288 C73GCK 56946617 IC50 > 100000 nM T11288 CL8Z0F 56946723 IC50 = 23300 nM T11288 CIQ64Z 56946724 IC50 = 17200 nM T11288 CXMK07 56946726 IC50 > 100000 nM T11288 CRY4C6 56946727 IC50 = 80000 nM T11288 CV29FO 56946728 IC50 > 100000 nM T11288 CI69QT 56946831 IC50 > 100000 nM T11288 CDPU29 56946832 IC50 > 100000 nM T11288 C69ELZ 56946833 IC50 = 6100 nM T11288 CH7M4O 56946835 IC50 > 100000 nM T11288 CP1VK5 56951135 IC50 > 200000 nM T11288 C1XCE9 57393400 IC50 > 100000 nM T11288 CJXP74 71061793 EC50 > 100000 nM T11288 CA2N0L 71062020 EC50 = 31800 nM T11288 C0QGU2 71062093 EC50 = 33200 nM T11288 C5T0NL 71454923 IC50 = 11180 nM T11288 C4ZD2W 71492590 IC50 = 418 nM T11288 C0P6IG 71492759 IC50 = 434 nM T11288 CV9QS7 71524587 EC50 > 100000 nM T11288 C7JIG6 71524588 EC50 > 100000 nM T11288 C1EY6B 71524589 EC50 = 14700 nM T11288 C4LPZ3 71524590 EC50 = 3200 nM T11288 C60ZQJ 71524591 EC50 = 8800 nM T11288 CGV8F5 71525288 EC50 > 100000 nM T11288 CO9ZJ3 71560809 EC50 > 100000 nM T11288 C0E6OM 71560810 EC50 > 100000 nM T11288 C3T8ZF 71560811 EC50 > 100000 nM T11288 CFN89Y 71560812 EC50 > 100000 nM T11288 C42SMF 71560938 EC50 > 100000 nM T11288 C98LPJ 71560939 EC50 > 100000 nM T11288 CG8DU1 71618156 EC50 > 100000 nM T11288 C0Z3PN 71682039 EC50 > 100000 nM T11288 CV5Z9M 71682040 EC50 > 100000 nM T11288 C1IZT7 71682041 EC50 > 100000 nM T11288 COV12T 71682195 EC50 > 100000 nM T11288 C3Y4FW 71682196 EC50 > 100000 nM T11288 CLF3I8 71682197 EC50 > 100000 nM T11288 CN6Q3L 71696716 EC50 = 113 nM T11288 CQCF98 71724480 EC50 = 151 nM T11288 C1PR7Z 71724504 EC50 = 140 nM T11288 CA7K8Z 71724506 EC50 = 217 nM T11288 CD9KH7 71724532 EC50 = 250 nM T11288 CWR2L5 71724556 EC50 = 220 nM T11288 C4ODQ2 71724557 EC50 = 425 nM T11288 C7T0UM 71724558 EC50 > 1000 nM T11288 CUL9E2 71724582 EC50 = 238.3 nM T11288 CNW68B 71724606 EC50 = 616.7 nM T11288 CCZ9B3 71724628 EC50 = 230 nM T11288 C48CAR 72735227 IC50 = 14090 nM T11288 CQ5NB6 72950792 IC50 = 21800 nM T11288 CF57OZ 73346145 IC50 = 19000 nM T11288 CK3EX6 73355255 IC50 = 27500 nM T11288 C7NTB0 73356802 IC50 = 15100 nM T11288 CRB93S 89784681 EC50 = 301.7 nM T11288 CG71EX 89784708 EC50 = 175 nM T11288 C4ZOX6 89784717 EC50 = 670 nM T11288 C0ZQO6 89784722 EC50 = 171 nM T11288 C4U5CZ 89784733 EC50 = 208 nM T11288 CW17YB 89784735 EC50 = 272 nM T11288 C0VD4P 89784742 EC50 = 114 nM T11288 CZT7B9 89784751 EC50 = 135 nM T11288 CH70XJ 89784752 EC50 = 193 nM T11288 C6MRA2 89784753 EC50 = 87 nM T11288 C1JH4L 89784756 EC50 = 243.3 nM T11288 CN1RD8 89784760 EC50 = 333.3 nM T11288 C2YB6Q 89784818 EC50 = 137 nM T11288 CSK8X6 89784827 EC50 = 233.3 nM T11288 CENX80 89785043 EC50 = 103 nM T11288 CY46QV 89785047 EC50 = 172.3 nM T11288 CQL7T6 89785059 EC50 = 99 nM T11288 CENR59 89785064 EC50 = 263 nM T11288 CVZG56 89785117 EC50 = 78 nM T11288 CT43OU 89785127 EC50 = 133.8 nM T11288 C3FB6Q 89785132 EC50 = 219 nM T11288 C4S9WG 89785146 EC50 = 650 nM T11288 CCE95J 89785148 EC50 = 184 nM T11288 C9SBA1 89785178 EC50 = 246.7 nM T11288 CSI51G 89785190 EC50 = 225 nM T11288 CGB2P5 89785210 EC50 = 276.3 nM T11288 CTY1H5 89785238 EC50 = 155 nM T11288 CHGX10 89785254 EC50 = 292.7 nM T11288 CB1FR2 89794901 EC50 = 441.7 nM T11288 C43AXK 89795130 EC50 = 750 nM T11288 C70LJV 89795278 EC50 > 1000 nM T11288 CFU4W2 89795305 EC50 = 760 nM T11288 CVB23M 89795326 EC50 = 245 nM T11288 CX1W9Z 89795330 EC50 = 165 nM T11288 C7XG4U 89795333 EC50 = 950 nM T11288 C7W1TP 89795335 EC50 = 475 nM T11288 CAX9S0 89795337 EC50 = 457.5 nM T11288 COB3Z9 89795340 EC50 = 180 nM T11288 C6BW0Q 89795341 EC50 = 137.7 nM T11288 CUHC90 90469229 EC50 = 11900 nM T11288 C05JQB 90469230 EC50 = 7000 nM T11288 C41EMT 90469289 EC50 = 3900 nM T11288 CA1VH0 90469291 EC50 = 12400 nM T11288 C4NX2Q 90469293 EC50 = 6600 nM T11288 C0NW8T 90469355 EC50 = 5200 nM T11288 C8BRG2 101876951 EC50 = 1100 nM T11288 C0H9DF 101891699 EC50 = 23000 nM T11288 CXHQ89 102340685 IC50 = 4280 nM T11288 CJ7VI3 102340686 IC50 = 6260 nM T11288 CS1P5K 102340687 IC50 = 3380 nM T11288 C93SXK 102340688 IC50 > 100000 nM T11288 C86WSC 117777746 EC50 = 255 nM T11288 C9E0BT 117777811 EC50 = 135 nM T11288 C9YPJ7 117803128 EC50 = 579 nM T11288 C5GUV9 118708511 IC50 = 5800 nM T11288 CQLK93 118708512 IC50 > 100000 nM T11288 C5F8LY 118708513 IC50 = 13600 nM T11288 CL8H6M 118708514 IC50 > 100000 nM T11288 CCT4I2 118708515 IC50 > 100000 nM T11288 C7GI8W 118708516 IC50 > 100000 nM T11288 CE7Q3U 118708517 IC50 > 100000 nM T11288 C31MGA 118708518 IC50 > 100000 nM T11288 CKV6P1 118708519 IC50 > 100000 nM T11288 C1MJ4N 118708520 IC50 > 100000 nM T11288 C7WFJ3 118708521 IC50 = 2200 nM T11288 CVK89G 118708522 IC50 > 100000 nM T11288 C7G3ZV 118708523 IC50 = 94500 nM T11288 CG8S9M 118708524 IC50 = 15800 nM T11288 C9T4KE 118708525 IC50 = 11100 nM T11288 CG3LK4 118708526 IC50 = 8130 nM T11288 C42ETW 118708527 IC50 = 23600 nM T11288 C0OQ9P 118716252 EC50 = 41400 nM T11288 C3VRT8 118716258 EC50 = 5200 nM T11288 C4Z2DS 118719365 EC50 = 10000 nM T11288 CU6EP1 122179376 IC50 = 322 nM T11288 CIL20J 122179390 IC50 = 142 nM T11288 C0OUW1 122179391 IC50 = 141 nM T11288 CCE46L 126587406 EC50 > 1000 nM T11288 CZG92F 127028059 IC50 = 11300 nM T11288 CSR0Y7 127028060 IC50 > 100000 nM T11288 C8Z2XI 127028354 IC50 = 19800 nM T11288 C8Q9DG 127028355 IC50 = 20800 nM T11288 CRI72H 127028356 IC50 = 22700 nM T11288 C58QBI 127028357 IC50 > 100000 nM T11288 C6AIP3 127028358 IC50 > 100000 nM T11288 CG46ES 127028359 IC50 = 30100 nM T11288 CRP9U1 127028361 IC50 = 53300 nM T11288 CUC9I4 127040367 IC50 = 18500 nM T11288 C0I9VF 127040368 IC50 = 5500 nM T11288 CX9JE1 127040369 IC50 = 8300 nM T11288 CRM9W5 127040370 IC50 = 1800 nM T11288 CJY60W 127042304 IC50 = 58300 nM T11288 CO2P8K 127042305 IC50 = 26700 nM T11288 C56HDS 127042306 IC50 = 8300 nM T11288 CRI0X9 127042307 IC50 > 100000 nM T11288 CK4J8D 127042801 IC50 = 7300 nM T11288 C87PMI 127042802 IC50 = 13200 nM T11288 CRQ7U8 127042918 IC50 = 10900 nM T11288 CDL84X 127042919 IC50 > 100000 nM T11288 C39PWZ 127042920 IC50 = 38000 nM T11288 C21DSU 127042921 IC50 = 6800 nM T11288 C6UZ7C 127042922 IC50 > 100000 nM T11288 CSBM31 127042943 IC50 = 12100 nM T11288 C12BJD 127042944 IC50 = 18800 nM T11288 CZBJ54 127048170 IC50 = 1010 nM T11288 CO93BJ 127048171 IC50 = 8980 nM T11288 C6L0AF 127049502 IC50 = 636 nM T11288 CK1SN3 127049508 IC50 = 1070 nM T11288 CB9EV4 127049509 IC50 = 2500 nM T11288 C7PF5I 127050480 IC50 = 623 nM T11288 C59EXD 127050481 IC50 = 876 nM T11288 CUO40Y 127050796 IC50 = 910 nM T11288 C7MJ5X 127050797 IC50 = 586 nM T11288 CT6A2G 127050798 IC50 = 2360 nM T11288 C6V7JZ 127051981 IC50 = 418 nM T11288 C4P0LG 127051982 IC50 = 821 nM T11288 C5CX0B 127051983 IC50 = 200 nM T11288 CBQL62 127051984 IC50 = 340 nM T11288 C0FOG1 127051985 IC50 = 866 nM T11288 C1VP2D 127052887 IC50 = 9410 nM T11288 CG9TE5 127052888 IC50 = 643 nM T11288 CA7N9R 127052889 IC50 = 981 nM T11288 C6ZK3C 135449697 EC50 > 100000 nM T11288 CD2NR8 136110930 IC50 = 95000 nM T11288 C1EB8Q 136236384 EC50 > 100000 nM T11288 CI0KU2 137643961 IC50 = 15900 nM T11288 CHCB46 145956407 IC50 = 44200 nM T11288 C1F4LH 145971569 IC50 > 1000 nM T11288 CK61NI 145973976 IC50 > 1000 nM T11288 CF8L7A 145979103 EC50 = 298 nM T11288 C3EX7W 145979504 EC50 = 170 nM T11288 C4G7LT 145980033 EC50 = 95 nM T11288 C26OWY 145981942 EC50 = 156 nM T11288 C13VFZ 145985646 EC50 = 53 nM T11288 C4A1LN 145985882 EC50 = 38000 nM T11288 CI38SJ 145987174 EC50 = 28900 nM T11288 CFU24J 145987833 EC50 = 103 nM T11288 CGL02K 145988126 EC50 = 205 nM T11288 CX3YR7 145990226 EC50 = 200 nM T11288 CZRB08 145990960 EC50 = 62000 nM T11288 CN1V8K 145992500 EC50 = 208 nM T11288 CT02XU 145992768 EC50 = 121 nM T11288 CKZA78 145992770 IC50 = 12500 nM T11288 C07OTB 145993028 EC50 = 111 nM T11288 C65JUT 145993130 EC50 > 1000 nM T11288 C3UC5J 145994097 EC50 = 207.3 nM T11288 CKM79V 145994277 EC50 = 155.8 nM T11288 C5VRT4 155511477 IC50 > 100000 nM T11288 C1L0WJ 155511549 IC50 = 20000 nM T11288 CE4C1X 155512695 IC50 = 5800 nM T11288 C0AFT8 155514623 EC50 > 1000 nM T11288 CH6O3X 155515825 EC50 = 5080 nM T11288 CV9TF6 155516191 EC50 > 1000 nM T11288 C4IS7E 155518051 EC50 = 2200 nM T11288 CLQO05 155518383 IC50 = 9680 nM T11288 CA1BD2 155520579 EC50 = 12700 nM T11288 C8WFN9 155522227 IC50 > 100000 nM T11288 C8V3OE 155522345 IC50 > 100000 nM T11288 CQK86M 155522385 IC50 > 100000 nM T11288 CS18PU 155523410 EC50 = 5600 nM T11288 CN6ST7 155523417 EC50 > 1000 nM T11288 C86ZPR 155525910 EC50 = 4400 nM T11288 C8TQ4G 155526547 EC50 > 1000 nM T11288 C9BGT5 155528240 EC50 > 1000 nM T11288 C75OQS 155529248 IC50 = 2980 nM T11288 C3O4FR 155529325 IC50 > 100000 nM T11288 C56AHP 155530068 EC50 = 181.4 nM T11288 C9F3YI 155530680 IC50 = 44000 nM T11288 C6I0LU 155531567 IC50 = 18000 nM T11288 CUL2G4 155531672 EC50 > 1000 nM T11288 CJ5X8R 155532908 IC50 = 322 nM T11288 C4IW9M 155533366 EC50 = 5800 nM T11288 C9QT4A 155533532 IC50 = 85100 nM T11288 CHF7A6 155535686 EC50 > 1000 nM T11288 C28CPM 155536187 IC50 = 3600 nM T11288 CQC9E5 155536529 IC50 > 100000 nM T11288 CGM43D 155536878 IC50 = 40000 nM T11288 CYG84N 155537154 EC50 = 7300 nM T11288 C2J7TM 155537461 IC50 = 17300 nM T11288 CGD47O 155537584 EC50 > 1000 nM T11288 CNS83Y 155538210 IC50 = 33000 nM T11288 CVES34 155538494 EC50 = 1900 nM T11288 CLU37N 155539307 EC50 = 3000 nM T11288 CXN6C4 155539538 IC50 = 31000 nM T11288 CL6QG0 155542981 IC50 = 73000 nM T11288 C7JUC3 155543680 EC50 = 4500 nM T11288 C1HI5E 155550141 IC50 > 100000 nM T11288 CB8FC1 155550293 EC50 = 3500 nM T11288 C8B3LI 155551011 IC50 = 3700 nM T11288 CX43TI 155551742 IC50 = 41000 nM T11288 CIF4T8 155553306 EC50 > 1000 nM T11288 CEZ7B1 155554618 EC50 = 137 nM T11288 CX6CM0 155554919 EC50 = 530 nM T11288 CU9P0W 155555392 IC50 = 18000 nM T11288 C7JI4C 155555932 EC50 = 348.3 nM T11288 C27XQN 155558615 EC50 = 212 nM T11288 C8ATZ5 155558917 IC50 = 53000 nM T11288 CUNV65 155558919 EC50 > 1000 nM T11288 CFRS42 155559312 IC50 > 100000 nM T11288 CG6NC7 155560071 EC50 = 10100 nM T11288 CE6C4X 155562808 IC50 > 100000 nM T11288 CWM67C 155563340 EC50 = 2800 nM T11288 C6Z2XK 155566234 EC50 = 3700 nM T11288 CO1LU7 155567143 EC50 > 1000 nM T11288 C7KFG6 155567619 EC50 = 3900 nM T11288 CTV5K3 155568177 EC50 > 1000 nM T11288 C03SJY 155568508 EC50 = 139.3 nM T11288 CTXV81 155568869 EC50 > 1000 nM T11288 C0K1HQ 155569340 IC50 = 12900 nM T11288 D00RFY 5281612 IC50 = 3000 nM T11288 D00RIX 5280443 Ki = 2400 nM T11288 D01FGM 5280666 IC50 = 3000 nM T11288 D07NAY 5281692 Ki = 5000 nM T11288 D0G3TK 5280863 Ki = 2400 nM T11288 D0I7GE 11790 IC50 = 11300 nM T11288 D0T3PW 5281672 Ki = 2400 nM T43115 CSI0D4 355 IC50 = 200000 nM T43115 CD6SZ4 69748 IC50 > 500000 nM T43115 CD42MV 94948 IC50 = 500 nM T43115 C0AVF1 95759 IC50 = 4100 nM T43115 C5X1YU 160254 IC50 = 41400 nM T43115 CV8A4D 163098 IC50 = 1000 nM T43115 C0C6FI 253328 IC50 = 4900 nM T43115 C8OHY9 254021 IC50 = 400 nM T43115 CZ91AU 315458 IC50 = 1200 nM T43115 CQ0LD7 344131 IC50 > 30000 nM T43115 CYZ86W 352335 IC50 = 800 nM T43115 CONR62 444765 Ki = 53000 nM T43115 C9B3YM 444766 Ki = 59000 nM T43115 CM0IQ3 446665 IC50 = 198000 nM T43115 C5Y3DJ 446871 Ki = 489000 nM T43115 CJ4M3B 448021 IC50 = 50000 nM T43115 CW5YV0 448024 IC50 = 50000 nM T43115 CHX62Y 598522 IC50 = 4500 nM T43115 C19XWM 1435211 IC50 > 90000 nM T43115 CC49RF 1450182 IC50 = 11000 nM T43115 CRC9X4 1902393 IC50 = 9700 nM T43115 CFK5Z0 2765033 IC50 = 79000 nM T43115 CQOC30 2765069 IC50 > 120000 nM T43115 CIV1E3 2775086 IC50 > 500000 nM T43115 CR8U7V 3182456 IC50 = 87000 nM T43115 CSIG03 3217106 IC50 = 90000 nM T43115 C9G0CA 3653077 IC50 = 10000 nM T43115 C12CHL 4470793 Ki > 300000 nM T43115 C8SZY6 4584157 IC50 > 100000 nM T43115 C35LZP 4774445 Ki = 41000 nM T43115 CPM09B 5327156 IC50 > 500000 nM T43115 CH5OM1 5463917 IC50 = 34200 nM T43115 C0PCZ3 5932584 IC50 = 500 nM T43115 CU65JT 5998084 IC50 = 610 nM T43115 C14LAC 6161281 IC50 = 460 nM T43115 CR6O8V 6166563 IC50 = 1800 nM T43115 CYI5R1 6274486 IC50 = 300 nM T43115 C3EI9B 6441564 IC50 > 30000 nM T43115 CZU0N8 7158830 IC50 > 100000 nM T43115 CPE73S 9547959 Ki = 26000 nM T43115 C54DXC 9813198 IC50 = 11000 nM T43115 C51LCY 9814234 IC50 = 7900 nM T43115 C3FP1L 9816159 IC50 = 38000 nM T43115 CQT1A6 9848618 IC50 > 50000 nM T43115 C54CTK 9863756 IC50 = 280 nM T43115 C86MNV 9864366 Ki = 1400000 nM T43115 CWIJ57 9873352 IC50 = 69000 nM T43115 C4BE0F 9874843 IC50 = 6300 nM T43115 C9XA0I 9895792 IC50 > 50000 nM T43115 C2JCM5 9902742 IC50 = 600 nM T43115 C6YF5L 9918081 Ki > 3000 nM T43115 CX91DJ 9920809 IC50 = 7000 nM T43115 CXD2Y6 9926586 IC50 = 200 nM T43115 CNA12K 9942558 IC50 = 1500 nM T43115 CSBA84 9966189 IC50 = 5500 nM T43115 CA75NG 9985013 IC50 = 42000 nM T43115 CO7T0B 10009840 IC50 > 50000 nM T43115 C6C9DL 10055263 Ki > 300000 nM T43115 CT64NM 10077494 IC50 = 1700 nM T43115 CF83UC 10094446 IC50 = 4100 nM T43115 C3Y8QT 10119338 IC50 = 5500 nM T43115 CPES42 10146934 IC50 = 25000 nM T43115 CSO2C9 10168739 IC50 = 50000 nM T43115 C0URF3 10169038 IC50 = 50000 nM T43115 CZ8JC5 10212468 IC50 = 50000 nM T43115 CHV18Y 10248262 IC50 = 600 nM T43115 CFQZ83 10252345 IC50 = 700 nM T43115 C3A8JL 10256983 IC50 = 14000 nM T43115 CN6D1Y 10267704 IC50 = 7700 nM T43115 C0O6CP 10305270 IC50 = 50000 nM T43115 CC30ZA 10305301 Ki > 200000 nM T43115 CZ90BA 10325640 IC50 > 19000 nM T43115 CX1YP3 10332717 IC50 > 1000000 nM T43115 C0D9QX 10372989 Ki > 30000 nM T43115 CS7DJ9 10404797 IC50 = 400 nM T43115 C5T0GC 10422621 IC50 > 1000000 nM T43115 C4J8LM 10433041 IC50 = 8500 nM T43115 C05SVE 10444314 IC50 = 3270 nM T43115 CZ50LG 10485602 IC50 = 50000 nM T43115 C30GDP 10491069 IC50 = 500 nM T43115 CFQ4G1 10493936 IC50 = 700 nM T43115 CKE4I0 10499065 IC50 = 600 nM T43115 C2TYE0 10499446 IC50 = 500 nM T43115 C70HFK 10509519 IC50 = 1100 nM T43115 CJKC18 10509653 IC50 = 1400 nM T43115 C95SPB 10509654 IC50 = 700 nM T43115 CIE96L 10509655 IC50 = 1000 nM T43115 CY93MH 10513846 IC50 = 840 nM T43115 C6Q0HE 10515600 IC50 = 22000 nM T43115 CK5F4M 10517813 IC50 = 800 nM T43115 C2U1ZS 10518152 IC50 > 30000 nM T43115 C3L1RU 10526652 IC50 = 5400 nM T43115 C8GX4H 10545864 IC50 = 800 nM T43115 CUMJ96 10556814 IC50 = 1100 nM T43115 CNM2H3 10556825 IC50 = 1400 nM T43115 CGN23O 10556999 IC50 = 800 nM T43115 C89LBE 10557509 IC50 = 600 nM T43115 CF5L2D 10582477 IC50 = 3700 nM T43115 C0DQ8N 10582552 IC50 = 800 nM T43115 C5EO4L 10582711 IC50 = 700 nM T43115 C3LAH0 10592371 IC50 = 3600 nM T43115 CYU34X 10605105 IC50 = 700 nM T43115 C5WZ8Y 10605302 IC50 = 900 nM T43115 CW45BF 10605499 IC50 = 700 nM T43115 C0QJ7S 10605667 IC50 = 1300 nM T43115 C9X3AT 10628013 IC50 = 600 nM T43115 CO1IZ0 10628864 IC50 = 1000 nM T43115 C1WR6S 10629318 IC50 = 1100 nM T43115 COLI53 10632854 IC50 > 30000 nM T43115 CV01CB 10638595 IC50 = 500 nM T43115 C1GFA2 10667311 IC50 = 1000 nM T43115 CJ7U3O 10668284 IC50 = 500 nM T43115 CZTN01 10675368 IC50 = 9100 nM T43115 CG3Q8I 10676936 IC50 = 600 nM T43115 C4UM9E 10700244 IC50 = 900 nM T43115 C5EV7N 10715582 IC50 = 700 nM T43115 CTY04W 10723912 IC50 = 1400 nM T43115 CUIW58 10723994 IC50 = 600 nM T43115 C5HE9F 10739445 IC50 = 1100 nM T43115 C15RHJ 10755924 IC50 = 800 nM T43115 C31IOZ 10757624 IC50 = 1000 nM T43115 CRC5Y3 10770793 IC50 = 900 nM T43115 C5UMR4 10771154 IC50 = 900 nM T43115 CC2U6K 10771506 IC50 = 1100 nM T43115 CPO6M5 10778347 IC50 = 8000 nM T43115 CEQD87 10782484 IC50 = 1000 nM T43115 CK9J4E 10783699 IC50 = 1200 nM T43115 C9XI7T 10804795 IC50 = 800 nM T43115 C1CNY2 10805901 IC50 = 3700 nM T43115 CIQB15 10818644 IC50 = 1900 nM T43115 C0TS2R 10843466 IC50 = 900 nM T43115 CJ1A6P 10854418 IC50 = 400 nM T43115 CT4H0O 11006141 IC50 = 108000 nM T43115 C2WP1J 11343454 IC50 = 22000 nM T43115 COIR53 11456678 IC50 = 5700 nM T43115 CRPL64 11516963 IC50 = 28800 nM T43115 C3P1EW 11702273 Ki > 1250000 nM T43115 C6A1LM 11786814 Ki = 77000 nM T43115 CV6K2W 11796020 IC50 > 100000 nM T43115 C6FUV5 11800375 IC50 = 12900 nM T43115 CWO5A6 11803410 IC50 = 1100 nM T43115 C9XF1H 12346155 IC50 = 8700 nM T43115 CZRS59 12394151 IC50 = 2300 nM T43115 C1L7WF 12678912 IC50 = 400 nM T43115 CN7H1V 12973096 IC50 = 1000 nM T43115 CE8Y4G 13779016 IC50 = 207100 nM T43115 C4KW7G 14024697 IC50 = 50000 nM T43115 CDJP28 15322751 IC50 = 3070 nM T43115 CL5H7V 15322752 IC50 = 5000 nM T43115 C0S5BD 15322755 IC50 = 2900 nM T43115 CRH5W9 15485891 IC50 = 19000 nM T43115 CKPF01 15485898 IC50 = 17000 nM T43115 CGQ81X 16046117 Ki = 33000 nM T43115 C0P4TQ 16220825 IC50 > 1000000 nM T43115 C17KIT 16220826 IC50 > 1000000 nM T43115 C0XZV4 16220827 IC50 > 1000000 nM T43115 CMX13P 16221752 IC50 > 1000000 nM T43115 C2PT9M 16221754 IC50 > 1000000 nM T43115 CM65WP 16221756 IC50 > 1000000 nM T43115 CY83SR 16221757 IC50 = 14000 nM T43115 C94LBM 17759043 Ki = 151000 nM T43115 C5TE6K 18398682 IC50 > 50000 nM T43115 CBQO20 18398709 IC50 > 50000 nM T43115 CJ4P9E 18957696 IC50 = 500000 nM T43115 CM1X6H 19350328 IC50 = 1000 nM T43115 C12GAZ 21145366 Ki > 30000 nM T43115 CH91UW 21265708 IC50 > 50000 nM T43115 CLI13Y 21265715 IC50 > 50000 nM T43115 C40CYN 21265722 IC50 > 50000 nM T43115 C1OR3D 22084082 Ki = 20000 nM T43115 C8CM6X 23427285 IC50 > 16000 nM T43115 CR6X9Y 23646522 IC50 = 50000 nM T43115 C6NH3C 23646669 Ki = 64000 nM T43115 C7ER2Q 23646672 Ki = 55000 nM T43115 CS18TW 24857885 IC50 > 50000 nM T43115 CJCY62 25055680 IC50 > 50000 nM T43115 CLS6X2 25055681 IC50 > 50000 nM T43115 CWMV64 25056374 IC50 > 50000 nM T43115 CNS2U7 25056375 IC50 = 26800 nM T43115 CU59JO 25056378 IC50 > 50000 nM T43115 C9BET0 25056379 IC50 > 50000 nM T43115 CT0H3U 25056635 IC50 > 50000 nM T43115 CC2Q6Z 25056895 IC50 > 50000 nM T43115 CE8J2D 25056896 IC50 > 50000 nM T43115 C40QFI 25147702 IC50 > 100000 nM T43115 C09KZA 25262525 IC50 = 186000 nM T43115 C4WM9S 25262527 IC50 = 30000 nM T43115 C4KO9Y 44265540 IC50 > 50000 nM T43115 C73QKU 44265541 IC50 = 25000 nM T43115 CJ6HG2 44265546 IC50 > 50000 nM T43115 CF2L9H 44265570 IC50 > 50000 nM T43115 CJ5C0R 44265576 IC50 > 50000 nM T43115 CK1Q2C 44265649 IC50 > 50000 nM T43115 COD4L3 44265670 IC50 = 7200 nM T43115 CWTQ56 44265697 IC50 = 50000 nM T43115 C8D9TY 44265698 IC50 = 11000 nM T43115 CB1H0Y 44265797 IC50 = 50000 nM T43115 CNLW94 44265857 IC50 = 50000 nM T43115 C7JLB1 44265863 IC50 = 64000 nM T43115 CD79RG 44265874 IC50 = 30000 nM T43115 CJQE06 44265877 IC50 = 50000 nM T43115 CSM7R2 44265887 IC50 = 50000 nM T43115 C2ZHC1 44295739 IC50 = 300 nM T43115 C4IVB9 44296058 IC50 = 1500 nM T43115 CCE0J4 44296059 IC50 = 1100 nM T43115 CA6M0Q 44296066 IC50 > 30000 nM T43115 CDJ1S7 44301133 IC50 = 1650 nM T43115 CI6Z0Y 44309201 IC50 = 58000 nM T43115 C4W9GA 44323010 IC50 > 1000000 nM T43115 C87MDN 44323030 IC50 = 120000 nM T43115 C3FIJ2 44323040 IC50 = 380000 nM T43115 C2SV7H 44323067 IC50 = 80500 nM T43115 CF3R6Y 44336593 Ki > 30000 nM T43115 CYX40O 44344614 IC50 = 279000 nM T43115 CT20HY 44359237 Ki = 210000 nM T43115 C5YV1R 44359299 Ki = 260000 nM T43115 CLH29B 44380956 IC50 > 100000 nM T43115 CWZ2G9 44381072 IC50 = 9100 nM T43115 CX28MD 44406938 IC50 = 150 nM T43115 C4VO7S 44407055 IC50 = 1230 nM T43115 C6YP9J 44447193 IC50 = 100000 nM T43115 CUA4L1 44449556 IC50 > 50000 nM T43115 CVD65P 44449557 IC50 > 50000 nM T43115 C74NTL 44449558 IC50 > 50000 nM T43115 CJ1F2K 44449627 IC50 > 50000 nM T43115 CV8DL7 44449628 IC50 = 37800 nM T43115 CVZ04W 44449658 IC50 > 50000 nM T43115 CRJA86 44449698 IC50 = 50000 nM T43115 C2DBZ3 44578543 IC50 = 280 nM T43115 C1ULD8 45483667 Ki = 37000 nM T43115 C45AFN 46186815 Ki > 100000 nM T43115 C7YZA3 46228445 IC50 = 66700 nM T43115 CBJ7Z6 46228829 IC50 = 33000 nM T43115 CCX49G 46228871 IC50 = 32600 nM T43115 CE1M2T 46228921 IC50 = 6700 nM T43115 C83GCS 46882340 IC50 > 44000 nM T43115 C3A2BY 49796575 IC50 = 180000 nM T43115 CGYM23 49796578 Ki = 9000 nM T43115 CMA49Q 49796582 IC50 > 100000 nM T43115 C2IU1Z 49796692 IC50 = 236000 nM T43115 C7YPR2 49797154 IC50 = 126000 nM T43115 CZR0Y3 49797156 IC50 = 29000 nM T43115 C4V3AU 49797169 IC50 = 280000 nM T43115 C4AEZ1 50925509 IC50 = 1050 nM T43115 C95QWO 50925510 IC50 = 410 nM T43115 CK1YX2 50941649 IC50 = 16200 nM T43115 C1PJL0 50941745 IC50 = 681 nM T43115 CRF1O3 50942131 IC50 = 877 nM T43115 CR8MG3 52947425 Ki = 40000 nM T43115 C93LZF 54682873 IC50 = 1200 nM T43115 CZ83RW 54751676 IC50 = 73000 nM T43115 CON5G1 54751677 IC50 = 81000 nM T43115 C9MP3W 54751678 IC50 > 100000 nM T43115 CCK72T 54751679 IC50 = 70000 nM T43115 C7K4GA 54757715 IC50 = 90000 nM T43115 C0NM6I 54757716 IC50 = 40000 nM T43115 CPX4I2 54757717 IC50 > 120000 nM T43115 C5OK3S 54757809 IC50 > 120000 nM T43115 C0DO1G 54757810 IC50 = 60000 nM T43115 CK49WP 54757811 IC50 = 80000 nM T43115 C5AQ8R 54757812 IC50 > 120000 nM T43115 CSPR73 54757813 IC50 > 120000 nM T43115 CK6Z3T 54757904 IC50 = 21000 nM T43115 C96NIW 54757905 IC50 > 100000 nM T43115 CT43AJ 54757906 IC50 = 33000 nM T43115 C93VEA 54758002 IC50 = 14000 nM T43115 C86LHU 54758003 IC50 = 2700 nM T43115 C79UJG 54758004 IC50 > 100000 nM T43115 C30WXK 54758005 IC50 = 2900 nM T43115 C2BT9H 70673568 IC50 = 12000 nM T43115 C3AJ7H 70981706 IC50 = 4200 nM T43115 CP4H6L 70981726 IC50 = 4100 nM T43115 C2KS7Y 70982811 IC50 = 3600 nM T43115 CXI0F3 71561559 IC50 > 100000 nM T43115 CE0Y3O 71561685 IC50 = 13000 nM T43115 C3M4CF 71561686 IC50 = 10000 nM T43115 C82KCZ 71561687 IC50 = 9000 nM T43115 CDA8P2 71561688 IC50 > 100000 nM T43115 C87EXF 71561689 IC50 = 5500 nM T43115 CP9HX5 71561815 IC50 = 900 nM T43115 C9H5YS 71561816 IC50 = 13100 nM T43115 C61MWP 71561817 IC50 = 11600 nM T43115 C9GO5M 71561818 IC50 = 120000 nM T43115 CWA30F 71561819 IC50 = 10100 nM T43115 CBC4G0 71561820 IC50 = 18900 nM T43115 CPV8Y3 71561944 IC50 = 14200 nM T43115 CPWU40 71597177 IC50 = 80000 nM T43115 CT4MK9 71717989 IC50 > 100000 nM T43115 CCY15D 71734765 IC50 = 3200 nM T43115 CMC9L2 72190151 IC50 = 8400 nM T43115 CKH70I 72705451 Ki > 500000 nM T43115 CCR34M 73345730 IC50 = 700 nM T43115 CX2KV0 73345731 IC50 = 1400 nM T43115 C1QYF5 73345732 IC50 = 900 nM T43115 CGU90Y 73350312 IC50 = 700 nM T43115 C24CNE 73351821 IC50 = 700 nM T43115 CM1W6X 73352369 IC50 = 59000 nM T43115 CFIB95 73353298 IC50 = 2000 nM T43115 CL8R6K 73354809 IC50 = 1800 nM T43115 CWJ6U5 73354810 IC50 = 800 nM T43115 CC1YW0 73354811 IC50 = 1000 nM T43115 CLSR90 73356355 IC50 = 1100 nM T43115 CSW01E 73356356 IC50 = 1200 nM T43115 C19JKD 101884098 IC50 > 100000 nM T43115 CO8V1Q 134130829 IC50 > 20000 nM T43115 C9BH3S 134131790 IC50 = 112400 nM T43115 C3Q6HX 134132029 IC50 > 20000 nM T43115 COG29Y 134132248 IC50 = 6600 nM T43115 CXM14Y 134132344 IC50 = 29100 nM T43115 CY4N3A 134132971 IC50 = 10900 nM T43115 CJV5H9 134133280 IC50 = 7800 nM T43115 CQV2R8 134133435 IC50 = 7600 nM T43115 CIM15P 134134309 IC50 > 500000 nM T43115 CK1ED4 134137535 IC50 > 20000 nM T43115 CO69VN 134138834 IC50 > 500000 nM T43115 C9WV1I 134139428 IC50 > 20000 nM T43115 CCS63E 134140312 IC50 = 3400 nM T43115 CFVU60 134141414 IC50 = 16100 nM T43115 C4E0TR 134148396 IC50 > 20000 nM T43115 C9NU1K 134148434 IC50 = 157200 nM T43115 CRG1A0 134150611 IC50 > 20000 nM T43115 CR72FZ 134152023 IC50 = 14900 nM T43115 C1FGJ5 134152452 IC50 = 5200 nM T43115 CO24SI 134154614 IC50 > 20000 nM T43115 C5CU3J 134157618 IC50 > 20000 nM T43115 CN23HD 134157879 IC50 = 2800 nM T43115 CBU6I2 137643274 IC50 > 27000 nM T43115 D07REK 343759 IC50 = 2000 nM T43115 D0E0BU 444763 Ki = 56000 nM T43115 D0F5VY 94860 IC50 = 2400 nM T43115 D0N7VL 52949968 Ki = 16000 nM T43115 D0Q2YJ 6763 IC50 = 700 nM T43115 D0SJ2Q 10494 IC50 = 1000 nM T43115 D0W9VA 10667 IC50 = 3000 nM T43115 D0Y1RO 1829 Ki = 49000 nM T43115 D0Y5SB 444764 Ki = 160000 nM T16808 D05EAM 4735 IC50 = 81000 nM T16808 D0U3YU 34755 IC50 = 12000 nM T16808 D0H2UB 5361 IC50 = 18100 nM T16808 CEXU05 3383 IC50 = 75000 nM T16808 CK4N7S 6293 IC50 = 1160000 nM T16808 C7MHL3 7009 IC50 = 540000 nM T16808 C0B2EX 10303 IC50 = 440000 nM T16808 CU14SM 11037 IC50 = 1220000 nM T16808 CH91QR 11049 IC50 = 1400 nM T16808 C1U2MY 12448 IC50 = 280000 nM T16808 CSI8A7 15785 IC50 = 1063000 nM T16808 CDMO72 18640 IC50 = 16300 nM T16808 CX94YJ 27020 IC50 = 1000 nM T16808 C5P3TH 65130 IC50 = 52000 nM T16808 C2IEY9 67062 IC50 = 227800 nM T16808 CM2RK5 67254 IC50 = 1200 nM T16808 CWU8N7 67338 IC50 = 39000 nM T16808 CWN04J 70420 IC50 = 126000 nM T16808 C1N7RQ 87052 IC50 = 1500 nM T16808 CQ8A5W 91330 Ki = 1710 nM T16808 CL4I5M 103900 IC50 = 68200 nM T16808 C0O3TQ 126437 IC50 = 9400 nM T16808 CS4X2H 208621 IC50 = 65600 nM T16808 CP6NH3 234402 IC50 = 1700 nM T16808 C0J1YF 246663 IC50 = 6100 nM T16808 CZI52L 409402 IC50 = 35400 nM T16808 C6SR4F 423583 IC50 = 56500 nM T16808 C1P4UJ 438070 IC50 = 1050000 nM T16808 CXU3P4 777039 IC50 < 20000 nM T16808 CU5TE7 833539 IC50 = 26700 nM T16808 CHQ4W1 847754 IC50 = 49700 nM T16808 CN7S8Q 850964 IC50 = 89000 nM T16808 CO49QA 969932 IC50 < 20000 nM T16808 C93NRD 988871 IC50 = 14100 nM T16808 CQEF34 1002773 IC50 > 100000 nM T16808 C34BFU 1098894 IC50 = 30400 nM T16808 C8G4OE 1192043 IC50 > 100000 nM T16808 CGK6Y1 1729769 Ki = 8400 nM T16808 CK09MX 2246814 IC50 = 205900 nM T16808 CV62YL 2297766 IC50 = 1029000 nM T16808 C58BST 2735117 IC50 = 885000 nM T16808 C89ATQ 2779831 IC50 = 12000 nM T16808 C52WEN 2827034 IC50 = 325000 nM T16808 CC94ZO 2829313 IC50 = 18900 nM T16808 CEZM97 2856635 IC50 = 234100 nM T16808 C5PRC6 3102693 IC50 = 1458000 nM T16808 C8RQO4 3246448 IC50 = 76100 nM T16808 CQM87H 3342878 IC50 = 519000 nM T16808 CSM6W2 3663787 IC50 = 70700 nM T16808 CG8F2A 3683950 Ki = 11300 nM T16808 CV2FS8 3899814 IC50 = 5000 nM T16808 C61VML 4110983 IC50 = 48900 nM T16808 CI3BC4 4334646 IC50 = 10200 nM T16808 C4TOJ7 4392904 IC50 = 43100 nM T16808 CH9K1U 5351747 Ki = 25600 nM T16808 CNK84Q 7128991 IC50 > 1000000 nM T16808 CG0D6N 10451940 IC50 > 100000 nM T16808 CEKH37 10979651 IC50 = 7200 nM T16808 CN3L1S 15883640 IC50 = 476000 nM T16808 CW6D8U 16116049 IC50 = 4800 nM T16808 CA1RW6 16116050 IC50 = 990000 nM T16808 CKU6L2 16212292 IC50 = 160800 nM T16808 CJ8H6E 16212367 IC50 = 284200 nM T16808 CBX8T9 16451230 IC50 = 37100 nM T16808 C4IAR3 16645216 IC50 > 100000 nM T16808 C94NBT 17756714 IC50 = 3000 nM T16808 CJQ86Y 24827559 IC50 > 667000 nM T16808 CJ4IC6 24962989 IC50 > 25000 nM T16808 CB3W4G 25086576 Ki = 4790 nM T16808 C7S1QA 25216415 IC50 > 100000 nM T16808 CR8F9X 25218467 IC50 > 100000 nM T16808 CI3D9O 30449576 IC50 = 867400 nM T16808 C0Y9FH 43199381 IC50 = 48000 nM T16808 CE52XJ 44420641 IC50 = 529000 nM T16808 C1A5UM 44420643 IC50 > 164000 nM T16808 CO20WN 44422923 IC50 = 54800 nM T16808 C2PT6B 46866514 IC50 = 95000 nM T16808 CHJ6C2 46868969 IC50 = 2370 nM T16808 C0N1JB 46884759 IC50 = 6200 nM T16808 C52HVN 46884802 IC50 = 2900 nM T16808 CUWR69 46884804 IC50 = 5600 nM T16808 CKAI31 53361222 IC50 > 667000 nM T16808 CV25JZ 53361223 IC50 > 667000 nM T16808 C0C6YK 53363652 IC50 > 667000 nM T16808 CPU86Z 53363653 IC50 > 667000 nM T16808 C63DVR 53363743 IC50 > 667000 nM T16808 COBL07 53363744 IC50 > 667000 nM T16808 C8QFS7 53363745 IC50 > 667000 nM T16808 CEG3P9 53363834 IC50 > 667000 nM T16808 CW4CD0 53363835 IC50 > 667000 nM T16808 C02ORV 53377508 Ki > 20000 nM T16808 CYM2T4 53868701 IC50 > 13000 nM T16808 CPL71I 54596764 IC50 > 100000 nM T16808 C6PRY0 56589655 IC50 = 3900 nM T16808 C72GHW 56642706 IC50 > 100000 nM T16808 CS6Q7R 56642708 IC50 > 100000 nM T16808 C2XR4C 56673504 IC50 = 11800 nM T16808 C3XKD4 56676677 IC50 = 45900 nM T16808 CV8A4S 56676725 IC50 = 6000 nM T16808 CP3MO9 56683405 IC50 = 68100 nM T16808 CY0IL9 56683483 IC50 = 35100 nM T16808 CJBY70 56951879 Ki > 50000 nM T16808 C04KFR 60150359 IC50 = 9500 nM T16808 CS8CJ7 66572090 IC50 = 6300 nM T16808 C60IYA 66572093 IC50 = 2560 nM T16808 CFID04 66572095 IC50 = 14300 nM T16808 C6L2RQ 66572097 IC50 = 368300 nM T16808 CFQ21S 66572099 IC50 = 291700 nM T16808 CER5F1 67466175 IC50 > 100000 nM T16808 C8JTS3 70676140 Ki > 100000 nM T16808 CZL47S 70676141 Ki > 100000 nM T16808 C8KC6O 70676142 Ki > 100000 nM T16808 CAFU69 70686225 IC50 = 4100 nM T16808 CH2C9T 70688341 IC50 = 20300 nM T16808 CN39YI 70692532 IC50 = 15500 nM T16808 C7QPK1 70694583 IC50 = 12000 nM T16808 C9CRO8 71583544 IC50 = 25200 nM T16808 CMW2X0 72947897 IC50 = 1810 nM T16808 CBK3U0 73892806 IC50 = 13000 nM T16808 CUP4Q6 76328021 Ki > 50000 nM T16808 CX7V5M 76328022 Ki > 50000 nM T16808 C5P2BM 76331683 Ki > 50000 nM T16808 C4XJ5N 78357767 IC50 > 100000 nM T16808 C9H7US 90667164 Ki = 2680 nM T16808 CE45VR 90667165 Ki = 2980 nM T16808 C23REW 90667166 Ki = 4290 nM T16808 CHT74V 90667167 Ki = 7620 nM T16808 CXSN29 90667168 Ki = 2900 nM T16808 C2YU1O 90667169 Ki = 2680 nM T16808 CQE25T 90667170 Ki = 7600 nM T16808 C73LWN 92136227 IC50 = 4 nM T16808 COA1W3 117666088 IC50 = 14 nM T16808 C5L8HT 118731724 IC50 = 1150 nM T16808 CWR35B 118731730 IC50 = 1250 nM T16808 CG83ZK 118731732 IC50 = 610 nM T16808 C0IT4N 118731735 IC50 = 6430 nM T16808 C2A8GF 118731737 IC50 = 2670 nM T16808 CWG18C 118731739 IC50 = 2030 nM T16808 CC96XD 118731741 IC50 = 4000 nM T16808 CI1AE0 118731742 IC50 = 3050 nM T16808 C6Y8BM 118731746 IC50 = 3380 nM T16808 CU0TW2 118731748 IC50 = 3390 nM T16808 CT3QY6 118731751 IC50 = 5760 nM T16808 CT1EF9 122195092 IC50 = 38000 nM T16808 C29SZC 122195093 IC50 = 9300 nM T16808 CRO3J8 122195094 IC50 = 13000 nM T16808 CIOL82 122195095 Ki = 1700 nM T16808 CE2BJ7 122195096 IC50 = 25000 nM T16808 C6KV9H 124081151 IC50 > 100000 nM T16808 C2GC5B 134144476 IC50 > 16000 nM T16808 CMHQ35 134153978 IC50 > 5800 nM T16808 CQ0ZO4 135308826 IC50 = 31 nM T16808 C5Y7GU 135406014 IC50 = 280600 nM T16808 CI8O9E 135967904 IC50 = 96000 nM T16808 CDXJ59 136180348 IC50 = 4200 nM T16808 C5PA4F 137169069 IC50 = 4000 nM T16808 CD1LT2 137633297 IC50 = 14000 nM T16808 C75JXU 137633379 IC50 = 14000 nM T16808 C4LK1X 137635057 IC50 > 50000 nM T16808 C20DYX 137644627 IC50 = 8200 nM T16808 C8NY6C 137644982 IC50 = 17000 nM T16808 CAP9N5 137652036 IC50 = 14000 nM T16808 CPA85Q 137655751 IC50 = 14000 nM T16808 CDPN65 137661881 IC50 > 50000 nM T16808 CR5D4S 138753329 IC50 = 5600 nM T16808 C51ILK 138753330 IC50 = 170 nM T16808 C8LEV4 139267760 IC50 > 10000 nM T16808 CE58DF 153041236 IC50 > 100000 nM T16808 CC50SM 155511980 IC50 = 58800 nM T16808 C1UAN2 155520348 IC50 = 20000 nM T16808 C7C8HI 155529624 IC50 = 8600 nM T16808 C67JQV 155538900 IC50 > 200000 nM T16808 CJ8ZI6 155549992 IC50 = 15000 nM T16808 D00FLT 65482 IC50 < 1000 nM T16808 D00SSW 6868 IC50 = 928000 nM T16808 D02TVQ 71268957 IC50 > 100000 nM T16808 D05UWW 23656549 IC50 = 55400 nM T16808 D09AFM 88489 IC50 = 8800 nM T16808 D09CLP 439155 Ki = 400 nM T16808 D0A0YX 5143 IC50 > 510000 nM T16808 D0BU8W 44219611 IC50 > 25000 nM T16808 D0Q3FY 44622850 IC50 > 25000 nM T86057 D07XGR 3339 IC50 > 75000 nM T86057 D0C3SW 53465279 IC50 = 6700 nM T86057 D0L7FM 4911 IC50 = 15000 nM T86057 D0NF1U 64929 IC50 = 11000 nM T86057 D0Z3DY 2333 IC50 = 22 nM T86057 D0O7QA 46840946 IC50 = 3500 nM T86057 D0P3ZN 54767229 IC50 = 23 nM T86057 D02JOK 86282507 IC50 = 58 nM T86057 D03UNB 86294127 IC50 = 33 nM T86057 D0HG2S 86294663 IC50 = 12 nM T86057 C1Y0DR 255968 IC50 = 2800 nM T86057 CU3FR4 2442078 IC50 = 1970 nM T86057 CA4F0Q 4480369 IC50 = 3610 nM T86057 CV5JP7 5089083 IC50 = 616 nM T86057 CF05JX 8193067 IC50 = 119 nM T86057 CX3Y5W 8193807 IC50 = 166 nM T86057 CK5Z9E 8500917 IC50 = 1970 nM T86057 C0DBP6 10320994 IC50 = 138 nM T86057 C2BF0Q 31071578 IC50 = 20 nM T86057 C42TZM 31809103 IC50 = 1480 nM T86057 CORM30 40175340 IC50 = 3920 nM T86057 CN97TL 40664355 IC50 = 1170 nM T86057 CPZI78 41529829 IC50 = 18 nM T86057 CFV19L 41529875 IC50 = 81 nM T86057 C0MU6Y 43091033 IC50 = 156 nM T86057 CY1AJ0 44547163 IC50 = 80 nM T86057 C6JL7F 52952152 IC50 = 2460 nM T86057 C10UTH 52952154 IC50 = 2490 nM T86057 CL2QX0 52952155 IC50 = 6680 nM T86057 CZT2O3 52952158 IC50 = 33650 nM T86057 CTP7V1 52952247 IC50 = 3920 nM T86057 C3D4SF 52952249 IC50 = 1130 nM T86057 CFJ5M9 52952250 IC50 = 19690 nM T86057 C6TA3F 52952361 IC50 = 3940 nM T86057 CI57AN 52952362 IC50 = 42 nM T86057 CSJ37V 52952363 IC50 = 189 nM T86057 C8X0KO 52952364 IC50 = 358 nM T86057 CZ70JQ 52952365 IC50 = 83 nM T86057 CWR97P 52952366 IC50 = 1440 nM T86057 CP0QO5 52952367 IC50 = 287 nM T86057 C2B6AK 52952469 IC50 = 111 nM T86057 C24YUT 52952470 IC50 = 1650 nM T86057 CPVA23 52952471 IC50 = 177 nM T86057 C2G3BJ 52952472 IC50 = 23460 nM T86057 CMO60U 52952473 IC50 = 667 nM T86057 C35UFW 52952474 IC50 = 772 nM T86057 CGQ72E 54764149 IC50 < 50 nM T86057 CM31TV 54767228 IC50 < 50 nM T86057 CU62OT 60596500 IC50 = 484 nM T86057 CY3FZ1 63000023 IC50 = 183 nM T86057 C1Q4UL 65661372 IC50 = 89 nM T86057 C7RNQ3 71973511 IC50 > 10000 nM T86057 CZL23E 86271138 IC50 = 1 nM T86057 CT0B8C 86279861 IC50 = 448 nM T86057 C52TCQ 86282513 IC50 = 3358 nM T86057 CSR54Q 86282791 IC50 = 110 nM T86057 CB9DY1 86291609 IC50 = 333.4 nM T86057 C0WPE1 86291610 IC50 = 115.3 nM T86057 C72IYH 86291611 IC50 = 659.2 nM T86057 CV8X7O 86291612 IC50 = 680.2 nM T86057 CGM1U7 86291613 IC50 > 10000 nM T86057 CP0IK1 86291614 IC50 = 1787 nM T86057 CKP6I8 86291615 IC50 = 1257 nM T86057 CL3S7B 86291616 IC50 > 10000 nM T86057 CKT4W2 86291776 IC50 = 206 nM T86057 C7M2WK 86291817 IC50 = 2757 nM T86057 CQ7VU5 86291818 IC50 = 343.2 nM T86057 C8QBZ6 86291819 IC50 = 129.8 nM T86057 CW1F6Y 86291820 IC50 = 352.3 nM T86057 CZ2O9R 86291821 IC50 = 324.3 nM T86057 CO0K7G 86291977 IC50 = 57 nM T86057 CHU74E 86294126 IC50 = 61.2 nM T86057 CW8JO2 86294128 IC50 = 342.8 nM T86057 CQWZ80 86294129 IC50 = 206.9 nM T86057 CD7S2F 86294305 IC50 = 1189 nM T86057 C2Z9ON 86294306 IC50 = 158.8 nM T86057 C58RHB 86294307 IC50 = 358.7 nM T86057 C7YXH2 86294308 IC50 = 197.8 nM T86057 CBT4J3 86294309 IC50 = 926.4 nM T86057 CX3LM9 86294310 IC50 = 1932 nM T86057 CX3UA5 86294311 IC50 = 557.6 nM T86057 C2M1RG 86294509 IC50 > 10000 nM T86057 CZR21V 86294510 IC50 = 1886 nM T86057 CLYB85 86294511 IC50 > 10000 nM T86057 C4XID3 86294512 IC50 = 398.8 nM T86057 CT05DV 86294514 IC50 = 1753 nM T86057 C2FL5M 117653246 IC50 = 37 nM T86057 CU87XO 117653280 IC50 = 92 nM T86057 CV9KA0 117653287 IC50 = 53 nM T86057 C3AV8J 117653356 IC50 = 19 nM T86057 CIRB95 117653498 IC50 = 74 nM T86057 CAHZ70 118009895 IC50 = 183 nM T86057 CJAD38 118009934 IC50 = 5147 nM T86057 C1RM8E 118009936 IC50 = 115 nM T86057 CHK1Y7 118009937 IC50 = 1823 nM T86057 CO68PR 118009938 IC50 = 1954 nM T86057 CEZ23L 118009939 IC50 = 395 nM T86057 C2V6YF 118009940 IC50 = 2982 nM T86057 CI60XP 118009944 IC50 = 382 nM T86057 C1CO5D 118009945 IC50 = 3868 nM T86057 CON28W 118010038 IC50 = 244 nM T86057 CM59EQ 118917669 IC50 = 42 nM T86057 C6J8YF 118917671 IC50 = 36 nM T86057 CQ24US 118917672 IC50 = 32 nM T86057 CY08KE 118934788 IC50 = 35 nM T86057 CL1XF2 124348595 IC50 = 127 nM T86057 CY9P8K 124570298 IC50 = 71 nM T86057 CV5P8R 125467587 IC50 = 111 nM T86057 CS5PN2 125467696 IC50 = 23 nM T86057 C67PLX 127038576 IC50 > 10000 nM T86057 C4QGW2 127041237 IC50 > 10000 nM T86057 CQL4H2 127041545 IC50 > 10000 nM T86057 C4T8DH 127042190 IC50 > 10000 nM T86057 CNB4R1 127042547 IC50 > 10000 nM T86057 CEP40Q 129323325 IC50 = 39 nM T86057 CYP1N5 129402245 IC50 = 18 nM T86057 CP5F6Q 129402246 IC50 = 199 nM T86057 CI9VE3 129402247 IC50 = 81 nM T86057 CVI62P 129402272 IC50 = 187 nM T86057 CHK1T7 129506542 IC50 = 29 nM T86057 CYZ80S 134136397 IC50 = 88 nM T86057 CXAN84 134137036 IC50 = 89 nM T86057 C2OLH1 134138549 IC50 > 10000 nM T86057 CUML27 134142855 IC50 = 1030 nM T86057 CZ6O8W 134147906 IC50 = 1123 nM T86057 C4LI8K 134152463 IC50 = 426 nM T86057 CZP0Q3 134154096 IC50 = 7 nM T86057 C2KH0W 134157756 IC50 = 185 nM T86057 C1SF0E 137631411 IC50 = 713 nM T86057 CH6D1A 137633664 IC50 = 4059 nM T86057 C7RLF8 137634145 IC50 = 1100 nM T86057 CA6P5N 137634324 IC50 = 215 nM T86057 CE3NQ4 137634953 IC50 = 9836 nM T86057 CU8LQ2 137635552 IC50 = 20900 nM T86057 C5NKL0 137641610 IC50 = 11999 nM T86057 CS1P3G 137642223 IC50 = 2000 nM T86057 CYF15J 137644133 IC50 = 2 nM T86057 C4LSW1 137644915 IC50 = 10 nM T86057 C94YSK 137648718 IC50 = 1400 nM T86057 C82IPK 137649192 IC50 = 241 nM T86057 C8E7MS 137649613 IC50 = 261 nM T86057 C9TU8I 137649663 IC50 = 390 nM T86057 CBWX69 137650724 IC50 = 3600 nM T86057 C4DXQ9 137653298 IC50 = 597 nM T86057 CN2X6I 137654849 IC50 = 2827 nM T86057 CDQ17K 137655704 IC50 = 4000 nM T86057 C95YOZ 137656797 IC50 = 127 nM T86057 CD86SW 137657077 IC50 = 203 nM T86057 C3KXD7 137662146 IC50 = 83 nM T86057 CMY7K5 138454759 IC50 = 32 nM T86057 CJR5H3 140870722 IC50 = 94 nM T86057 C1KWO4 155512239 IC50 = 10210 nM T86057 C6XJ4G 155518043 IC50 = 1660 nM T86057 CUMC45 155520477 IC50 = 1550 nM T86057 C5BAX4 155527014 IC50 = 280 nM T86057 CBTP61 155527375 IC50 = 365000 nM T86057 CR41AU 155532458 IC50 = 5100 nM T86057 C4I2RA 155533226 IC50 = 640 nM T86057 CM6A4W 155536773 IC50 = 5410 nM T86057 CZN6I0 155540397 IC50 = 6380 nM T86057 C26PMG 155540831 IC50 = 15780 nM T86057 CQ3BI2 155555487 IC50 = 10570 nM T86057 C3JU1A 155556604 IC50 = 2200 nM T86057 CLIA01 155557315 IC50 = 2790 nM T86057 C24FSC 155558289 IC50 = 3240 nM T86057 C2T3BD 155560602 IC50 = 14380 nM T86057 C41VAC 155563560 IC50 = 4050 nM T86057 CLPQ15 155567122 IC50 = 1940 nM T86057 C4WI2F 155569549 IC50 = 119000 nM T86057 D0NJ4H 5281670 IC50 = 2000 nM T87930 D00ENY 33032 Ki = 701 nM T87930 COC91V 10255 Ki = 8 nM T87930 C6T4AH 167842 Ki = 9.1 nM T87930 CO28NU 447407 EC50 = 480 nM T87930 C3JXD9 5289518 EC50 = 100 nM T87930 C5Z8VG 6324635 Ki > 10000 nM T87930 CVW4L3 9795654 Ki = 2.9 nM T87930 C2L6EK 9807075 Ki = 25000 nM T87930 C9TLQ4 9861035 Ki > 10000 nM T87930 CG0WB9 9958244 Ki = 20000 nM T87930 CRJ2T0 10219992 Ki = 10000 nM T87930 C5PD0H 10330442 Ki = 7500 nM T87930 C7GIJ3 10398361 Ki = 21400 nM T87930 CX1V3L 10437436 Ki = 12000 nM T87930 CXE7F5 10541731 Ki > 10000 nM T87930 CJZ04V 11096831 Ki = 393 nM T87930 CDGZ79 11820131 Ki = 82200 nM T87930 CLRK62 22097088 Ki = 1300 nM T87930 C0YK6J 22100077 Ki > 30000 nM T87930 CM9D7U 22100122 Ki = 18000 nM T87930 CJ8UB0 22100152 Ki = 9800 nM T87930 CIG65E 22449297 Ki = 11000 nM T87930 C4U7OS 44152410 Ki = 57.1 nM T87930 CJ5X0B 44307207 Ki = 20000 nM T87930 C1JC7K 44307264 Ki = 25000 nM T87930 C8U2SF 44307281 Ki > 30000 nM T87930 CW9TR7 44346780 Ki = 30.9 nM T87930 C64ELF 44346789 Ki = 1150 nM T87930 CQJW06 44346790 Ki = 1980 nM T87930 C15MPO 44346798 Ki = 19.8 nM T87930 D01DMS 447196 Ki = 0.24 nM T87930 D03NDD 9935648 Ki = 8900 nM T87930 D04SMQ 440053 Ki = 28900 nM T87930 D09LXQ 126569 Ki = 1820 nM T87930 D0KD6O 5288598 EC50 = 130 nM T87930 D0T5SU 158397 Ki = 2144 nM T74312 D00STL 644241 IC50 = 9548 nM T74312 D01PZD 5329098 IC50 = 160 nM T74312 D03ZBT 11626560 IC50 > 1000 nM T74312 D04AIT 5280445 IC50 = 830 nM T74312 D04KZY 49803313 IC50 = 0.29 nM T74312 D04LVK 57379345 IC50 = 60 nM T74312 D07NVU 9829523 IC50 = 30 nM T74312 D08PIE 68165256 IC50 = 2.1 nM T74312 D09GDD 11167602 IC50 = 82 nM T74312 D09KTS 24821094 IC50 > 1000 nM T74312 D0AZ3C 5291 IC50 = 131 nM T74312 D0E7PQ 5311 IC50 > 10000 nM T74312 D0H0EQ 24826799 IC50 = 0.3 nM T74312 D0IQ6P 25102847 IC50 = 6 nM T74312 D0J9ZR 4477 IC50 > 100000 nM T74312 D0K8KX 5280343 IC50 = 590 nM T74312 D0R0MW 5329102 IC50 = 3 nM T74312 D0V9WF 126565 IC50 = 1.5 nM T74312 D0W5HK 216239 IC50 = 1.3 nM T74312 D00ABO 11427553 IC50 = 6.6 nM T74312 D00DRL 44137946 IC50 = 22 nM T74312 D00RYA 16750271 IC50 = 60 nM T74312 D00UZR 5330286 IC50 = 3480 nM T74312 D01CNB 10172827 IC50 = 5 nM T74312 D02RJY 11442891 IC50 = 669 nM T74312 D02XNW 5494449 IC50 = 30 nM T74312 D03HUX 49792852 IC50 = 510 nM T74312 D03LWG 53235510 IC50 = 3252 nM T74312 D04PBH 5280804 IC50 > 10000 nM T74312 D05PZB 135398495 IC50 = 10 nM T74312 D06DMQ 59472121 Ki = 18 nM T74312 D06KTJ 53252276 IC50 = 4.6 nM T74312 D07EHV 44814409 IC50 > 10000 nM T74312 D07HPJ 11476171 IC50 = 1400 nM T74312 D07KYT 24889392 IC50 < 0.51 nM T74312 D08DHN 67286591 Ki > 4000 nM T74312 D08UUL 46700756 IC50 = 385.98 nM T74312 D09JEJ 24748573 IC50 = 55 nM T74312 D09TAB 25151352 IC50 = 5 nM T74312 D0CY1B 6420138 IC50 = 25.12 nM T74312 D0D1GF 42642645 IC50 = 3.6 nM T74312 D0E3TC 44259 IC50 = 0.52 nM T74312 D0FD6D 11751922 IC50 = 71 nM T74312 D0G8BM 16722836 IC50 = 15 nM T74312 D0G9AW 59473233 EC50 = 327 nM T74312 D0J1GR 10366136 IC50 = 3 nM T74312 D0M9QZ 11485656 IC50 = 5 nM T74312 D0O0LS 25141092 IC50 = 164 nM T74312 D0O6WV 24794418 IC50 = 16 nM T74312 D0P0KN 16739650 IC50 = 21 nM T74312 D0P1CV 46191454 IC50 > 10000 nM T74312 D0PN8H 46216796 IC50 = 6 nM T74312 D0Q7RE 16007391 IC50 = 100 nM T74312 D0S6TK 11213558 EC50 = 10 nM T74312 D0S7HM 16041424 IC50 = 1.86 nM T74312 D0SG7B 49831257 IC50 = 338 nM T74312 D0Z4RC 24756910 IC50 = 1500 nM T74312 D03BNU 59604787 IC50 > 3500 nM T74312 D01OLO 9820526 IC50 = 618 nM T74312 D06GBK 2048 IC50 = 1100 nM T74312 D09HEV 6539952 IC50 = 24 nM T74312 D0H4GI 10275001 IC50 = 1.6 nM T74312 D0IT6Q 3038522 IC50 = 33 nM T74312 D0T3ME 156422 IC50 > 30000 nM T74312 C97TNH 10177 IC50 > 10000 nM T74312 C63WLY 89644 IC50 = 4.8 ug.mL-1 T74312 C5JE2Z 104860 IC50 = 0.66 ug.mL-1 T74312 CZC9W3 124286 IC50 = 4722 nM T74312 CI1NA5 159926 IC50 = 0.85 ug.mL-1 T74312 CYBA43 177458 IC50 = 2.5 ug.mL-1 T74312 CLF3D2 403163 IC50 = 10070 nM T74312 C75HBM 403164 IC50 = 212 nM T74312 CH20NR 403176 IC50 = 418 nM T74312 CR0TC3 425532 IC50 > 2000 nM T74312 C7HME8 439246 IC50 > 10000 nM T74312 C76DPL 667885 IC50 = 560 nM T74312 CTY2J9 667938 IC50 = 170 nM T74312 C4C6LE 673481 IC50 = 1300 nM T74312 CG2H9B 673603 IC50 = 52 nM T74312 CE85VC 675676 IC50 > 10000 nM T74312 C6DX3A 675881 IC50 = 120 nM T74312 C1J6ZU 675892 IC50 > 10000 nM T74312 CGP4Y9 678521 IC50 = 2000 nM T74312 CW19EP 678543 IC50 = 3200 nM T74312 C49GDM 678544 IC50 = 360 nM T74312 C9JL0R 679570 IC50 > 10000 nM T74312 C71MCT 681617 IC50 = 3600 nM T74312 C3CDV9 690904 IC50 = 140 nM T74312 C3KG7U 704777 IC50 = 630 nM T74312 C5O8CZ 722715 IC50 = 1100 nM T74312 C5LCA8 722862 IC50 = 3000 nM T74312 C24FKL 723132 IC50 = 250 nM T74312 C1XP4H 723141 IC50 > 10000 nM T74312 C1AEV3 747044 IC50 > 10000 nM T74312 C48NVR 764010 IC50 = 110 nM T74312 C9HE2Z 794754 IC50 = 2100 nM T74312 C7AZV0 831009 IC50 = 140 nM T74312 CECK45 841038 IC50 = 140 nM T74312 CB27WS 849733 IC50 > 10000 nM T74312 C7MOF3 874463 IC50 = 1000 nM T74312 CC7GK6 961926 IC50 = 110 nM T74312 C9CI5M 984977 IC50 = 630 nM T74312 CF0JO3 1035391 IC50 > 10000 nM T74312 CI54DH 1074680 IC50 = 1700 nM T74312 C7EO6D 1083543 IC50 = 250 nM T74312 CI5U8L 1083545 IC50 = 490 nM T74312 CIY4M3 1086009 IC50 = 10000 nM T74312 CJR18A 1112313 IC50 = 310 nM T74312 CW74PK 1181875 IC50 = 130 nM T74312 CGV40B 1505876 IC50 = 443 nM T74312 C81BFU 1742780 IC50 > 100000 nM T74312 CP69TN 2059507 IC50 > 10000 nM T74312 C62PLI 2066142 IC50 = 310 nM T74312 CEBT92 2171072 IC50 = 6900 nM T74312 CJ2S8E 2225147 IC50 = 27 nM T74312 CHC5I0 2971839 IC50 > 10000 nM T74312 CFY1D0 2974957 IC50 > 10000 nM T74312 CF97WY 3392650 IC50 = 590 nM T74312 CA3C5S 3685259 IC50 < 5000 nM T74312 CJ96CI 4042130 IC50 = 2700 nM T74312 CG12IM 4378773 IC50 > 10000 nM T74312 CDBS50 4799247 IC50 = 281 nM T74312 C8UH5F 5162557 IC50 = 540 nM T74312 C23WZE 5320315 IC50 = 1480 nM T74312 C4RUV5 5329453 IC50 = 1 nM T74312 CDQ3M7 5359485 IC50 = 0.43 ug.mL-1 T74312 C54BYP 5360741 IC50 = 1 ug.mL-1 T74312 C3XIO2 5718145 IC50 > 12500 nM T74312 CUPQ08 6539985 IC50 = 2 nM T74312 CMEZ23 6540005 IC50 = 27 nM T74312 CK19HQ 6540021 IC50 = 10 nM T74312 CXK07R 6540022 IC50 = 59 nM T74312 CFLH24 6540023 IC50 = 140 nM T74312 CJ17TA 6540024 IC50 = 67 nM T74312 C0BQ2E 6540025 IC50 = 700 nM T74312 CIUP42 6540026 IC50 = 130 nM T74312 CFYE71 9341021 IC50 = 417 nM T74312 C4MW6D 9411754 IC50 = 310 nM T74312 CJ1ML3 9412007 IC50 = 352 nM T74312 CQ8HP2 9413573 IC50 = 552 nM T74312 CX10KR 9828962 IC50 = 70 nM T74312 CBGE59 9833337 IC50 = 5300 nM T74312 CHF7G5 9890746 IC50 = 14900 nM T74312 C3EUB4 9911005 IC50 = 3300 nM T74312 C1BZ0P 9928737 IC50 = 14 nM T74312 CW8VZ6 9950868 IC50 = 3810 nM T74312 C91SZV 9966132 IC50 = 640 nM T74312 CUJR40 10062694 EC50 > 2000 nM T74312 C5WCL2 10117540 IC50 = 450 nM T74312 C3ER4N 10187285 IC50 = 8790 nM T74312 CD7J3O 10231458 IC50 = 100 nM T74312 CAE03L 10231813 IC50 = 128 nM T74312 CC4G8B 10302519 IC50 = 1910 nM T74312 C4FP8M 10303591 IC50 = 200 nM T74312 C6ZF0X 10386217 IC50 = 7020 nM T74312 CMO39Z 10405910 Ki = 24 nM T74312 C1GBL0 10427414 Ki = 42 nM T74312 C7HBP6 10429593 IC50 > 10000 nM T74312 C95LYF 10457505 IC50 = 11400 nM T74312 C9ELW2 10754937 IC50 > 30000 nM T74312 C47NIR 10801110 IC50 = 5800 nM T74312 CJ4P5T 10905857 IC50 = 19700 nM T74312 CJ05CL 11048367 IC50 = 50 nM T74312 C03XHM 11152545 IC50 = 4 nM T74312 CW6Z5P 11154134 IC50 = 10 nM T74312 CB47NS 11156401 IC50 = 34 nM T74312 C6KMU2 11176194 IC50 = 8 nM T74312 CU53KH 11177394 IC50 = 1570 nM T74312 C7ZB5L 11177668 IC50 = 106 nM T74312 CNG8F1 11178869 IC50 = 215 nM T74312 C6H5VA 11189551 IC50 = 27 nM T74312 CM1L0D 11203646 IC50 = 2 nM T74312 CSWR60 11223082 IC50 = 1500 nM T74312 CT0C5R 11235290 IC50 = 64 nM T74312 C8CF1H 11244819 IC50 = 54 nM T74312 C1Y7DB 11245809 IC50 = 14 nM T74312 CJFX60 11259128 IC50 = 13 nM T74312 CV18PX 11265647 IC50 = 619 nM T74312 CBQ10L 11268741 IC50 = 55 nM T74312 CQL3P9 11271710 IC50 = 24 nM T74312 CC24PZ 11281789 IC50 = 1260 nM T74312 CBOP58 11293798 Ki > 10000 nM T74312 C60ISR 11304968 IC50 = 213 nM T74312 CYK15J 11314310 IC50 = 12 nM T74312 CL7G8F 11325920 IC50 = 4 nM T74312 CY54IT 11337407 IC50 = 8 nM T74312 CK1P7Y 11337894 IC50 = 3 nM T74312 CUT16W 11340683 IC50 = 15 nM T74312 C26BZX 11362471 Ki > 10000 nM T74312 CY8AQ4 11371508 IC50 = 5 nM T74312 C25ZCN 11374110 IC50 = 19 nM T74312 CWXB93 11397177 Ki > 10000 nM T74312 CNT8W2 11404903 IC50 = 39 nM T74312 CPIM91 11406239 IC50 = 22 nM T74312 C6EP7S 11407183 IC50 = 8 nM T74312 CL7I5H 11407736 IC50 = 270 nM T74312 C6ML4B 11417108 IC50 = 157 nM T74312 CI34BN 11428396 IC50 = 25 nM T74312 C6LJR3 11429321 IC50 = 173 nM T74312 CREQ51 11429654 IC50 = 36 nM T74312 CY0A4E 11429729 IC50 = 30 nM T74312 C5KG7W 11440661 IC50 = 5 nM T74312 CAM63T 11451774 IC50 = 6 nM T74312 C2U9EF 11452379 IC50 = 270 nM T74312 CD97KV 11462058 IC50 = 7 nM T74312 CJ94MR 11465254 IC50 = 450 nM T74312 CN20YG 11465676 IC50 = 82 nM T74312 CJ2BH4 11473904 IC50 = 26 nM T74312 CK3M0T 11495270 IC50 = 2 nM T74312 CTRF08 11501874 IC50 > 30000 nM T74312 C93ZMH 11502131 IC50 = 10000 nM T74312 CRU9D3 11508262 Ki = 8 nM T74312 CEQC69 11509096 IC50 = 6700 nM T74312 C2T8YD 11511361 IC50 = 58 nM T74312 CKMX76 11514852 IC50 > 30000 nM T74312 CG3BZ9 11517980 IC50 = 7 nM T74312 C5KA2B 11530692 IC50 = 4.9 nM T74312 CL7X4Q 11530963 IC50 = 270 nM T74312 CTG83F 11539329 Ki > 2500 nM T74312 CAO2C1 11543838 IC50 = 4400 nM T74312 C6O8IK 11551046 IC50 = 2600 nM T74312 CD4XU0 11552138 IC50 = 3400 nM T74312 CVZG65 11558401 IC50 = 340 nM T74312 C7CBV5 11558574 IC50 = 6600 nM T74312 CACS26 11561968 Ki = 800 nM T74312 C98AHV 11573064 IC50 = 10000 nM T74312 CQOI76 11576375 IC50 = 450 nM T74312 CPW27V 11581044 Ki = 11 nM T74312 C4M1FH 11581469 IC50 = 9900 nM T74312 CO9KP5 11583459 IC50 > 10000 nM T74312 C13TED 11587554 IC50 = 2600 nM T74312 C3VUO7 11588815 IC50 = 4 nM T74312 CMK39C 11589776 IC50 = 1300 nM T74312 CB91RQ 11589811 IC50 = 80 nM T74312 CA2KX0 11590078 IC50 < 3 nM T74312 CM65QP 11590120 IC50 = 10 nM T74312 CMIL86 11590363 Ki > 2500 nM T74312 COQ86X 11594510 IC50 > 30000 nM T74312 CEN64F 11594651 IC50 = 10000 nM T74312 C8KYF4 11594711 IC50 = 10000 nM T74312 CV19LS 11594712 IC50 = 7600 nM T74312 C1TP3Q 11603793 IC50 = 36 nM T74312 C69FYK 11604142 Ki = 0.17 nM T74312 C43JZU 11604436 IC50 = 5000 nM T74312 CGU7N0 11604739 IC50 > 20000 nM T74312 CJU5W6 11611103 Ki = 69 nM T74312 C8IKG5 11616255 IC50 = 60 nM T74312 C9UCV6 11616461 IC50 = 10000 nM T74312 C9G2KW 11616810 IC50 > 30000 nM T74312 CQF4W9 11623433 IC50 = 740 nM T74312 CCO9Q6 11630723 IC50 = 1000 nM T74312 C7W3TE 11633427 IC50 = 20 nM T74312 CYL45U 11634544 IC50 = 8 nM T74312 C8V0YT 11639969 IC50 = 220 nM T74312 C35XTQ 11640048 IC50 = 1500 nM T74312 C9T6SC 11640926 Ki > 2500 nM T74312 CU3WZ7 11652264 IC50 = 170 nM T74312 C0XF6R 11652445 IC50 = 670 nM T74312 CQ4OC2 11654378 IC50 = 18 nM T74312 CAJS96 11662893 IC50 > 20000 nM T74312 C8GM0V 11666441 IC50 = 1200 nM T74312 C6UF8I 11666980 IC50 = 10000 nM T74312 CKAH36 11669784 IC50 = 4000 nM T74312 CMF26K 11673988 IC50 = 920 nM T74312 CVJO30 11681070 IC50 = 530 nM T74312 CJ9KN7 11683817 IC50 > 10000 nM T74312 CHG14R 11688408 IC50 = 9400 nM T74312 CU0E8O 11690457 Ki = 250 nM T74312 CRJW43 11702271 IC50 = 880 nM T74312 CB0AP2 11705863 Ki = 910 nM T74312 CFE7S4 11709608 IC50 = 11000 nM T74312 CE49IU 11718919 Ki = 120 nM T74312 CUB2N6 11719537 IC50 = 9 nM T74312 C9P0VD 11729539 IC50 > 30000 nM T74312 CU5V9K 11749082 IC50 = 17 nM T74312 C8MOK3 11750699 IC50 < 1000 nM T74312 CN6Z7I 11751616 IC50 > 10000 nM T74312 CP7AH3 11755812 IC50 = 2000 nM T74312 CN1U7P 11855937 IC50 = 28 nM T74312 CYA0X2 11856199 IC50 = 22 nM T74312 C0A9WL 11856200 IC50 = 60 nM T74312 CJ5G9Y 11856201 IC50 = 37 nM T74312 COLP81 11856204 IC50 = 16 nM T74312 CSRQ05 11856467 IC50 = 61 nM T74312 CA2BL5 11856735 IC50 = 58 nM T74312 CW53JC 11998038 Ki = 100 nM T74312 CI39TK 12004372 IC50 = 50 nM T74312 CN81RQ 12004373 IC50 = 36 nM T74312 CRY1Z3 12004374 IC50 = 58 nM T74312 CG80CI 12004395 IC50 = 62 nM T74312 CGBO48 12004396 IC50 = 18 nM T74312 C4IJG5 12004397 IC50 = 3 nM T74312 CP4KW5 12004398 IC50 = 99 nM T74312 C6B9SJ 12004399 IC50 = 146 nM T74312 CJ90ZE 12375089 IC50 > 2000 nM T74312 CPV7R2 12440912 IC50 = 2300 nM T74312 CG95AZ 12440913 IC50 = 1700 nM T74312 C08UDR 13393482 IC50 > 30000 nM T74312 C0G5VS 13393483 IC50 > 30000 nM T74312 CY02TK 13393484 IC50 > 30000 nM T74312 CAG6O8 13454369 IC50 > 30000 nM T74312 CS3H4X 13714289 IC50 = 1400 nM T74312 C2SLB7 13714290 IC50 = 4400 nM T74312 CDGF78 15282555 IC50 = 2400 nM T74312 CQN23V 15551239 IC50 = 630 nM T74312 C24FXN 15941243 IC50 = 2696 nM T74312 CG5IO2 15941244 IC50 = 145 nM T74312 C8Y1XP 15941246 IC50 = 2 nM T74312 CB94LR 15941247 IC50 = 13 nM T74312 CZ38JG 15941390 IC50 = 135 nM T74312 CE57UJ 15941392 IC50 = 2 nM T74312 C1AIM6 15941393 IC50 = 16 nM T74312 CN7PO9 15941394 IC50 = 6 nM T74312 C9E3RP 15941395 IC50 = 7 nM T74312 CSBF70 15941529 IC50 = 9 nM T74312 CQM93O 15941530 IC50 = 3 nM T74312 CFPW41 16007116 Ki > 2500 nM T74312 C9JK2M 16059071 IC50 = 1 nM T74312 CW6UJ9 16059338 IC50 = 3 nM T74312 CH7MS6 16059729 IC50 = 1 nM T74312 COIK65 16070059 IC50 = 110 nM T74312 C1VQ0J 16124774 IC50 = 3 nM T74312 CX7FV0 16124775 IC50 = 26 nM T74312 CGF2M4 16124831 IC50 = 47 nM T74312 CU1K9R 16124836 IC50 = 860 nM T74312 C3FS0I 16124974 IC50 = 73 nM T74312 C3B8SQ 16124975 IC50 = 120 nM T74312 CD3U0I 16124976 IC50 = 34 nM T74312 C9R4EN 16125232 IC50 = 2 nM T74312 C9XMJ4 16125233 IC50 = 7 nM T74312 C4BFJ3 16125303 IC50 = 480 nM T74312 CZM0J2 16125381 IC50 = 29 nM T74312 CVAZ06 16125453 IC50 = 60 nM T74312 CP3HS4 16220354 IC50 = 9 nM T74312 CVZK29 16223008 IC50 = 120 nM T74312 C4TC3X 16722832 IC50 = 25 nM T74312 C0V8FB 16730091 IC50 > 800 nM T74312 CA24TE 16730092 IC50 > 1000 nM T74312 C4Q2TN 16739431 IC50 = 98 nM T74312 CWI96A 16739432 IC50 = 25 nM T74312 CSE35D 16739464 IC50 = 770 nM T74312 C20OFQ 16739508 IC50 = 120 nM T74312 CNFX02 16739511 IC50 = 77 nM T74312 C3AGL1 16739512 IC50 = 160 nM T74312 C0JTZ9 16739677 IC50 = 1000 nM T74312 C4IX1K 16739678 IC50 = 310 nM T74312 COZ7A1 16739706 IC50 = 270 nM T74312 C0HB9T 16739709 IC50 = 190 nM T74312 C0U8DY 16739710 IC50 = 40 nM T74312 COC6L0 16739741 IC50 = 2750 nM T74312 C1Z8WO 16739742 IC50 = 66 nM T74312 CPT2G0 16739743 IC50 > 10000 nM T74312 CPC5Q9 16739745 IC50 > 10000 nM T74312 CLY96T 16739777 IC50 = 42 nM T74312 C0TMW8 16739778 IC50 = 22 nM T74312 C1MAE7 16739807 IC50 = 1700 nM T74312 C9H8XT 16739808 IC50 > 10000 nM T74312 CC5UB1 16739809 IC50 = 2900 nM T74312 CQ43TS 16739810 IC50 = 30 nM T74312 CJCN32 16739811 IC50 > 10000 nM T74312 CDK6A4 16739812 IC50 = 140 nM T74312 CE0I5O 16739835 IC50 = 30 nM T74312 C4C7DF 16739839 IC50 = 71 nM T74312 C20BPQ 16739840 IC50 = 35 nM T74312 CE1XT6 16739866 IC50 = 1450 nM T74312 C8JBR9 16739867 IC50 = 250 nM T74312 C1VG0U 16739870 IC50 = 45 nM T74312 C2Z4DB 16739901 IC50 = 93 nM T74312 C1UFH7 16739902 IC50 = 110 nM T74312 C7DFM1 16739903 IC50 = 490 nM T74312 CHX86I 16739904 IC50 = 350 nM T74312 CCP56J 16739905 IC50 = 12 nM T74312 CP9C6B 16739918 IC50 = 440 nM T74312 CJB7M2 16739919 IC50 = 23 nM T74312 C2WNB4 16739920 IC50 = 19 nM T74312 CQ64XI 16739921 IC50 = 22 nM T74312 C9MT8U 16739933 IC50 = 150 nM T74312 CM3UF8 16739935 IC50 = 1200 nM T74312 CFEP56 16739948 IC50 = 310 nM T74312 CKE6V9 16739949 IC50 = 310 nM T74312 C23KZR 16739951 IC50 = 4800 nM T74312 C6GJ5Q 16739952 IC50 = 37 nM T74312 CFRU87 16739965 IC50 = 29 nM T74312 CDZ31W 16747696 IC50 = 22 nM T74312 C9OQ1G 16750272 IC50 = 620 nM T74312 CW2SY5 16750291 IC50 = 24 nM T74312 CIX7U2 16750304 IC50 = 48 nM T74312 C6A3XS 16750306 IC50 = 45 nM T74312 CB2TK1 16750327 IC50 = 180 nM T74312 CH4O1C 16750328 IC50 = 63 nM T74312 C90MJD 16750331 IC50 = 560 nM T74312 CTG1Y0 16866350 IC50 > 2000 nM T74312 CCM03E 16866353 IC50 > 2000 nM T74312 C1TK9R 16866354 IC50 = 786 nM T74312 C25UKC 21081761 IC50 = 4 nM T74312 CBD9U4 23647620 IC50 = 2600 nM T74312 C2RV3U 24180608 IC50 > 30000 nM T74312 C5CKW8 24752189 IC50 = 16 nM T74312 CA3I4T 24753787 IC50 > 50000 nM T74312 C0D2PA 24758868 IC50 > 1000 nM T74312 C3K5YO 24758982 IC50 > 1000 nM T74312 CYU0Z8 24758983 IC50 > 1000 nM T74312 CJL67N 24759089 IC50 > 20000 nM T74312 C2APK8 24759090 IC50 > 1000 nM T74312 C5CRF6 24759091 IC50 > 1000 nM T74312 CA8U7X 24759094 IC50 > 1000 nM T74312 CRB89L 24759205 IC50 > 1000 nM T74312 C13JUP 24759314 IC50 > 1000 nM T74312 C7YG1N 24759534 IC50 < 10 nM T74312 CQNP54 24764449 IC50 = 391 nM T74312 CCF17D 24768394 IC50 = 68 nM T74312 CYK71D 24768395 IC50 > 12500 nM T74312 C7EXG0 24768396 IC50 = 1400 nM T74312 CP1WR0 24795070 IC50 = 21 nM T74312 C5YW7P 24825755 IC50 = 1517 nM T74312 C9B2TF 24880043 IC50 = 6 nM T74312 CFK2B9 24882503 IC50 > 10000 nM T74312 C43HWQ 24883287 IC50 > 10000 nM T74312 C8DA5Q 24883334 IC50 > 10000 nM T74312 C4V9GH 24894117 IC50 = 6100 nM T74312 CM6K3X 24894768 IC50 = 44000 nM T74312 CJH19T 24894883 IC50 = 5000 nM T74312 CJ14YB 24894884 IC50 = 9900 nM T74312 CHVU39 24894885 IC50 = 14000 nM T74312 CZ6KD4 24894886 IC50 = 34000 nM T74312 CKBY19 24894887 IC50 = 25000 nM T74312 CB5TP8 24894992 IC50 = 20000 nM T74312 C32SUJ 24894993 IC50 = 36000 nM T74312 CP7QT2 24894995 IC50 = 2200 nM T74312 CF4N9X 24895100 IC50 = 3000 nM T74312 C0RVS3 24896719 IC50 = 133 nM T74312 CJ7XN5 24896721 IC50 = 175 nM T74312 CDHC95 24896725 IC50 = 540 nM T74312 C07EFA 24898056 IC50 = 69 nM T74312 CIGQ12 24898058 IC50 = 611 nM T74312 CU9P6M 24898062 IC50 = 750 nM T74312 CWC6F4 24898259 IC50 = 470 nM T74312 CP3M7W 24898267 IC50 = 175 nM T74312 CG51ON 24898486 IC50 = 65 nM T74312 CP27GV 24898487 IC50 = 1603 nM T74312 C78VZS 24898709 IC50 = 208 nM T74312 CO86UD 24899176 IC50 = 488 nM T74312 C3BT6M 24899425 IC50 = 546 nM T74312 CWV98O 24899557 IC50 = 93 nM T74312 CPN09F 24899684 IC50 = 78.71 nM T74312 CK37DA 24899686 IC50 = 47.08 nM T74312 CS76PW 24899690 IC50 = 721 nM T74312 C5T2KO 24899691 IC50 = 633 nM T74312 CN13JF 24899915 IC50 = 0.33 ug.mL-1 T74312 CBWR97 24899916 IC50 = 0.53 ug.mL-1 T74312 C9F2JD 24899917 IC50 > 10 ug.mL-1 T74312 C0NCB3 24899936 IC50 = 787 nM T74312 CG0TV5 24899942 IC50 = 301 nM T74312 C64MTI 24900160 IC50 = 1.8 ug.mL-1 T74312 CO2I6Q 24900161 IC50 = 6.6 ug.mL-1 T74312 CZ6S7L 24900183 IC50 = 91.23 nM T74312 CO3Z6U 24900185 IC50 = 282 nM T74312 C7E4HO 24900190 IC50 = 85 nM T74312 C5FD1A 24937369 IC50 = 36 nM T74312 C9YN2Q 24967131 IC50 > 10000 nM T74312 CS3Q8B 24995659 Ki = 580 nM T74312 C4KG0Y 25022599 IC50 = 47 nM T74312 CH90KV 25097876 IC50 = 2 nM T74312 C9L5ID 25098154 IC50 = 47 nM T74312 CAO38V 25098429 IC50 = 8 nM T74312 COV8Z0 25143021 IC50 > 10000 nM T74312 C6BWZ8 25145145 IC50 = 76 nM T74312 C78YWA 25145716 IC50 = 14 nM T74312 CI0E2L 25154395 IC50 = 31 nM T74312 CL1W5D 25154436 IC50 = 31 nM T74312 CIUJ83 25167109 IC50 = 448 nM T74312 COB9G8 25181586 IC50 = 41200 nM T74312 C76WYH 25184035 IC50 = 69 nM T74312 CX3F4U 25195515 IC50 = 55000 nM T74312 CNG96H 25210579 IC50 = 659 nM T74312 C8IJB9 25218207 IC50 = 39600 nM T74312 C2TXC6 25218656 IC50 = 41 nM T74312 CQ3LF1 25226298 IC50 = 642 nM T74312 CI9QX8 25264352 IC50 > 1000 nM T74312 CFP1U6 25264354 IC50 = 60 nM T74312 C4X7GK 40562736 IC50 > 10000 nM T74312 CU2B4F 42611245 IC50 = 132 nM T74312 C75GFD 42633960 Ki = 46 nM T74312 CJ5U1X 42639664 IC50 = 2.8 ug.mL-1 T74312 CA0E4U 44132585 IC50 = 14 nM T74312 CAK0F2 44155856 IC50 < 3 nM T74312 CD0YP3 44159001 Ki = 160 nM T74312 CUQE83 44187007 IC50 = 17 nM T74312 C8KNA3 44219632 Ki = 1400 nM T74312 C0VIX4 44219633 Ki = 2300 nM T74312 C0LDV8 44222965 IC50 = 70 nM T74312 C3ZJ6S 44222969 IC50 = 61 nM T74312 CX4SQ0 44222970 EC50 > 10000 nM T74312 CV1X8T 44256373 IC50 = 3.6 nM T74312 CF6SL7 44256410 IC50 = 4 nM T74312 CCOI94 44405868 IC50 = 900 nM T74312 CM5B3A 44405870 IC50 = 13700 nM T74312 C1VT7R 44417767 IC50 = 795 nM T74312 C51BYS 44420784 IC50 = 13 nM T74312 CW1V7M 44423636 IC50 = 270 nM T74312 CETQ79 44427518 IC50 > 50000 nM T74312 COPG94 44427519 IC50 > 10000 nM T74312 CP5MR0 44433459 IC50 = 50 nM T74312 COT78K 44433461 IC50 = 340 nM T74312 CPE5U4 44433462 IC50 = 75 nM T74312 CWC8V3 44433464 IC50 = 15 nM T74312 C6VB4Q 44433471 IC50 = 1370 nM T74312 CJ9UC7 44433472 IC50 = 1 nM T74312 CCT13U 44433473 IC50 = 14 nM T74312 CWP17E 44433506 IC50 = 150 nM T74312 CZQ21O 44433507 IC50 = 165 nM T74312 C6WMP3 44433508 IC50 = 41 nM T74312 C0AG3T 44433509 IC50 = 260 nM T74312 C65GTN 44433510 IC50 = 18 nM T74312 C4BOK8 44433511 IC50 = 49 nM T74312 CGV37F 44440254 IC50 = 153 nM T74312 C5JUV3 44440256 IC50 = 624 nM T74312 CFB56S 44440259 IC50 = 65 nM T74312 CEW9G2 44440261 IC50 = 1108 nM T74312 C13FIN 44450007 IC50 = 2858 nM T74312 CLK0W7 44453682 IC50 = 34 nM T74312 CYH6P3 44520205 IC50 = 1100 nM T74312 CL3M2Q 44545852 IC50 = 134 nM T74312 C6I1TW 44560803 IC50 = 5 nM T74312 CW2JN3 44589504 IC50 = 106 nM T74312 CA5HP8 44589505 IC50 = 4.8 nM T74312 CX6RQ2 44589506 IC50 = 34 nM T74312 CQZV09 44589507 IC50 = 80 nM T74312 CQ8RF5 44589837 IC50 = 373 nM T74312 CZH4E2 44590190 IC50 = 35 nM T74312 CUO2C8 44590191 IC50 = 63 nM T74312 CD8V7Q 44590192 IC50 = 515 nM T74312 CEK73Z 44590193 IC50 = 47 nM T74312 CI90QD 44590194 IC50 = 134 nM T74312 CU3RF1 45139989 IC50 > 10000 nM T74312 CQGZ06 45139991 IC50 > 10000 nM T74312 CNYA73 45482631 IC50 = 1740 nM T74312 CNI92D 46182735 IC50 = 2.3 nM T74312 CF57GK 46215462 IC50 = 0.9 nM T74312 CY3HW5 46224684 IC50 = 5900 nM T74312 CYT37A 46232443 IC50 = 46000 nM T74312 C48ZVW 46232555 IC50 = 32000 nM T74312 CS9B1U 46232556 IC50 = 15000 nM T74312 C85RJI 46233108 IC50 = 2300 nM T74312 C19SZF 46233185 IC50 = 400 nM T74312 C7ON5A 46233287 IC50 > 10000 nM T74312 C9H4YO 46233889 IC50 = 730 nM T74312 CRT34L 46235770 IC50 = 95 nM T74312 CBU6Y0 46830369 IC50 = 7 nM T74312 CJB36H 46869713 IC50 = 9 nM T74312 CQB16A 46872415 Ki > 4000 nM T74312 CLS29B 46872626 IC50 > 10000 nM T74312 CIZA86 46890251 IC50 = 96 nM T74312 CTZ71Y 46898039 IC50 = 0.5 nM T74312 CVQ3T8 46898068 IC50 = 25 nM T74312 CQLT07 46913878 IC50 < 1000 nM T74312 C2HZ3M 49779260 IC50 > 10000 nM T74312 CH5NU2 49798965 IC50 = 17.3 nM T74312 C02SVR 49798997 IC50 = 7.3 nM T74312 C8DA5K 49798998 IC50 = 97.8 nM T74312 CO18QM 49798999 IC50 = 51.2 nM T74312 CC8FS1 49799031 IC50 = 1.4 nM T74312 CLNI64 49799032 IC50 = 4 nM T74312 CG7K2D 49799066 IC50 = 1.2 nM T74312 C27SKR 49799067 IC50 = 0.9 nM T74312 CCX04I 49799068 IC50 = 1.9 nM T74312 CQZC18 49799069 IC50 = 0.8 nM T74312 C2HA1O 49799301 IC50 = 2.7 nM T74312 C62OBF 49799302 IC50 > 1000 nM T74312 C1QC4V 49799333 IC50 > 1000 nM T74312 CG3LY7 49799334 IC50 > 1000 nM T74312 CZBW04 49799372 IC50 = 0.7 nM T74312 CN1M2D 49799373 IC50 = 1.5 nM T74312 CHIQ50 49799374 IC50 = 0.2 nM T74312 C45FZO 49799375 IC50 = 14.9 nM T74312 CNL8F1 49799533 IC50 > 20000 nM T74312 CHSF07 49806372 IC50 > 1000 nM T74312 CB0S2P 49842666 IC50 = 330 nM T74312 C5R6QY 49842669 IC50 = 34000 nM T74312 C0NA9U 49842670 IC50 = 2500 nM T74312 CC7MR2 49842671 IC50 = 16000 nM T74312 CAI20B 49842778 IC50 = 330 nM T74312 CRA74I 49842779 IC50 = 850 nM T74312 CF91RS 49843531 IC50 > 10000 nM T74312 C7A6IZ 49850211 IC50 = 150 nM T74312 CBC62W 50899254 IC50 = 194 nM T74312 CQ3KU9 50899556 IC50 < 1 nM T74312 CK5TH3 50906783 IC50 = 890 nM T74312 CVQ6P3 50915164 IC50 > 10000 nM T74312 C2Y6QS 50938552 IC50 > 10000 nM T74312 CAZQ43 51003133 IC50 = 5 nM T74312 C5NT2O 51036049 IC50 > 10000 nM T74312 CK0MX5 51036250 IC50 = 5300 nM T74312 C9NYP4 51036677 IC50 > 10000 nM T74312 C4WRY3 51037112 IC50 > 10000 nM T74312 CDTC84 51037916 IC50 > 10000 nM T74312 CRI28Z 51037948 IC50 > 10000 nM T74312 CXA03W 52920796 IC50 = 46 nM T74312 C1VML8 52936434 Ki = 32 nM T74312 CU1T5C 52936530 Ki = 6 nM T74312 CK69ML 52936531 Ki = 5 nM T74312 CCT6B9 52936532 Ki = 20 nM T74312 CC7SE4 52936533 Ki = 80 nM T74312 CA93FM 52936534 Ki = 110 nM T74312 C9KO7D 52936535 Ki = 1045 nM T74312 CEQN27 52936621 Ki = 20 nM T74312 C2A6MX 52936622 Ki = 140 nM T74312 CBH0K9 52936623 Ki = 80 nM T74312 CKF2D5 52936624 Ki = 410 nM T74312 CM24LF 52938983 IC50 < 1 nM T74312 CC9F0Q 52941363 IC50 = 39 nM T74312 C7P9AL 52941426 IC50 > 1000 nM T74312 CX1S9K 52941548 IC50 = 14 nM T74312 C3LB5V 52941849 IC50 = 130 nM T74312 C2C8ZO 52942593 IC50 = 30 nM T74312 C6YG2W 52942653 IC50 > 1000 nM T74312 C1ETR0 52942740 IC50 = 5 nM T74312 C17JTA 52943859 IC50 = 90 nM T74312 CW2X5E 52944268 IC50 = 1 nM T74312 C8CVQ2 52944383 IC50 = 23 nM T74312 CQ6E9L 52944516 IC50 = 742 nM T74312 C3N9BD 52945116 IC50 = 86 nM T74312 CCS4Y6 52945585 IC50 > 1000 nM T74312 CSU36D 52945586 IC50 = 128 nM T74312 C6FXB2 52945601 IC50 = 350 nM T74312 C9PX2J 52945752 IC50 < 1 nM T74312 CL4ED3 52945753 IC50 = 1 nM T74312 C3LE5D 52945818 IC50 = 224 nM T74312 C71HRI 52946208 IC50 = 19 nM T74312 CGY30T 52946358 IC50 = 177 nM T74312 CVE40F 52946431 IC50 = 17 nM T74312 C24ZMH 52947505 IC50 > 1000 nM T74312 C3KH4N 52947592 IC50 = 18 nM T74312 CIR3Q0 52947964 IC50 = 120 nM T74312 CDI7W6 52948729 IC50 > 1000 nM T74312 COJ3H6 52949299 IC50 > 1000 nM T74312 CF2HT3 52949521 IC50 = 12 nM T74312 CVF59K 52949935 IC50 = 1460 nM T74312 CVC5K1 52950048 IC50 = 12 nM T74312 CJ56EO 53244398 IC50 = 18 nM T74312 C64IQX 53244399 IC50 >= 3000 nM T74312 C1P3BC 53244475 IC50 >= 1500 nM T74312 C8ZTF9 53249002 IC50 = 6692 nM T74312 C6OTY5 53251320 IC50 > 30000 nM T74312 C2P3OT 53316977 IC50 = 2400 nM T74312 CE8OY2 53317913 IC50 = 5 nM T74312 CX59LD 53320915 IC50 = 7100 nM T74312 CZY0J7 53323592 IC50 = 590 nM T74312 CCKD48 53324892 IC50 = 12000 nM T74312 CNPM14 53341082 IC50 > 3000 nM T74312 C8ZRE3 53356518 IC50 = 479 nM T74312 CE8OA7 53357593 IC50 = 6 nM T74312 CNI7P9 53372541 IC50 = 231 nM T74312 C0IYG7 53372543 IC50 > 1000 nM T74312 CA6H2P 53372668 IC50 = 125 nM T74312 CY1I9B 53372669 IC50 = 778 nM T74312 COP26H 53372670 IC50 = 12 nM T74312 CFM7W8 53372672 IC50 = 7000 nM T74312 C9GYZ3 53372790 IC50 = 4350 nM T74312 CVG4Q3 53379717 IC50 = 42.6 nM T74312 C8NA4L 53384644 IC50 > 30000 nM T74312 CVG90B 53389651 IC50 > 10000 nM T74312 CO6B0E 54583043 IC50 > 10000 nM T74312 C3PGE2 54585958 IC50 > 10000 nM T74312 CV7HJ8 54585959 IC50 > 10000 nM T74312 C8AB1J 54759606 Ki < 0.3 nM T74312 CBO2L1 54761157 IC50 = 1 nM T74312 CS23GM 54762055 IC50 = 2 nM T74312 CY3V6S 54764326 IC50 > 10000 nM T74312 C9EMO2 54765177 IC50 = 9.5 nM T74312 CXQ0R1 56593680 Ki = 5 nM T74312 C7O3DJ 56593681 Ki = 8 nM T74312 CSO49B 56593682 Ki = 5 nM T74312 CUQ2Z3 56593684 Ki = 12 nM T74312 CVT2Y9 56593685 Ki = 11 nM T74312 C6VOK1 56593686 Ki = 10 nM T74312 CIMU73 56593834 Ki = 12 nM T74312 CCVD67 56593835 Ki = 9 nM T74312 CZIM93 56593836 Ki = 2 nM T74312 C6V9LJ 56593837 Ki < 1 nM T74312 CUP6Z9 56593838 Ki = 5 nM T74312 C5T3NA 56595430 Ki = 85 nM T74312 CPT6H4 56595552 Ki = 22 nM T74312 CTM84F 56595553 Ki = 210 nM T74312 CQUH59 56595554 Ki = 11 nM T74312 CYEQ07 56595555 Ki = 2500 nM T74312 C6PXQ5 56595556 Ki = 930 nM T74312 C5BD6I 56595557 Ki = 53 nM T74312 C5KR6N 56595558 Ki = 2.8 nM T74312 COI9U2 56595687 Ki = 15 nM T74312 C2AM6B 56595688 Ki = 18 nM T74312 CFY2I4 56595689 Ki = 6 nM T74312 CAM8E1 56595690 Ki = 12 nM T74312 CN5EV7 56595691 Ki = 15 nM T74312 C6ET0W 56595693 Ki = 1 nM T74312 C9DX3J 56649281 IC50 = 12.22 nM T74312 CBZ8T4 56657856 IC50 = 226 nM T74312 CTR10F 56658543 Ki = 22 nM T74312 C8IZ4J 56659759 IC50 = 10 nM T74312 CPG0I4 56659823 IC50 = 160 nM T74312 C4UPH5 56659824 IC50 = 7 nM T74312 CVDT38 56659825 IC50 = 110 nM T74312 C3A7HL 56663233 IC50 = 10 nM T74312 CRQ78A 56663280 IC50 = 14 nM T74312 CY12ML 56663288 IC50 = 120 nM T74312 CK53GA 56663289 IC50 = 65 nM T74312 CY2RD1 56663290 IC50 > 1000 nM T74312 C6XVT5 56666663 IC50 = 50 nM T74312 CKE5U3 56666717 IC50 = 350 nM T74312 CDB0L7 56666718 IC50 = 270 nM T74312 CN25KP 56670130 IC50 > 1000 nM T74312 C1HTO5 56670140 IC50 = 100 nM T74312 CC3J1A 56673651 IC50 = 11 nM T74312 C4TD2Q 56673654 IC50 = 8 nM T74312 CYPL60 56675140 IC50 = 216 nM T74312 CGN54D 56676922 IC50 = 60 nM T74312 CU0M8W 56676973 IC50 = 7 nM T74312 CH5R3Q 56676974 IC50 = 15 nM T74312 CUD53B 56676975 IC50 = 29 nM T74312 C91XIW 56676976 IC50 = 20 nM T74312 CO2GI9 56676977 IC50 = 120 nM T74312 CL5HZ3 56680292 IC50 > 1000 nM T74312 CFS43O 56680303 IC50 = 590 nM T74312 C5RK1U 56680304 IC50 = 360 nM T74312 CJL83V 56682400 Ki = 7 nM T74312 CSX3Y4 56683569 IC50 = 71 nM T74312 CVM7U4 56683624 IC50 = 90 nM T74312 CBW28D 56683625 IC50 = 70 nM T74312 CR4H3M 56835099 IC50 = 9300 nM T74312 CP8T5I 56835100 IC50 = 1100 nM T74312 CY36EG 56945171 IC50 = 720 nM T74312 C4OG7H 56945172 IC50 = 970 nM T74312 CH0QA3 56945173 IC50 = 590 nM T74312 CM0NQ5 56945174 IC50 = 1600 nM T74312 CXKF03 56945175 IC50 = 5600 nM T74312 C6WU4V 56945277 IC50 = 28 nM T74312 C7D0EY 56946378 IC50 = 210 nM T74312 CUQ50W 56946379 IC50 = 140 nM T74312 CAK91L 56955954 IC50 > 3600 nM T74312 CPHX64 57325478 IC50 > 50000 nM T74312 CQ9BW4 57325479 IC50 > 50000 nM T74312 CPO2J4 57342178 IC50 = 73 nM T74312 C72PED 57342179 IC50 = 7.9 nM T74312 CA93PN 57342180 IC50 = 17 nM T74312 CU3WM8 57390291 IC50 = 103 nM T74312 CO92HZ 57390346 IC50 = 46 nM T74312 C4WE9B 57391179 IC50 = 4 nM T74312 CY10TP 57391180 IC50 = 4 nM T74312 CU3DM9 57391295 IC50 > 1000 nM T74312 CS27KY 57391922 IC50 = 6700 nM T74312 CIA26P 57391923 IC50 = 9700 nM T74312 CVO51K 57391924 IC50 = 10900 nM T74312 CT6E2B 57391925 IC50 = 10200 nM T74312 CG5LM0 57392126 EC50 = 2600 nM T74312 CZT5Q4 57392128 EC50 = 8900 nM T74312 CU7J9C 57393063 IC50 = 3 nM T74312 CD4HS3 57393074 IC50 = 8 nM T74312 CS60KL 57393075 IC50 > 800 nM T74312 C16RBI 57393424 IC50 = 58 nM T74312 CW4K5T 57393650 IC50 = 6300 nM T74312 CHG95S 57393892 EC50 = 4400 nM T74312 CKVG97 57394105 IC50 < 1000 nM T74312 CWMT98 57394785 IC50 > 1000 nM T74312 C9PY4Q 57394798 IC50 > 60 nM T74312 C3F9VS 57394799 IC50 > 400 nM T74312 C29ZPK 57395544 IC50 > 25000 nM T74312 C4CN6V 57396453 IC50 > 20 nM T74312 CCT58R 57396454 IC50 = 10 nM T74312 CXA5Z9 57396541 IC50 = 20 nM T74312 CPAH35 57396542 IC50 = 4 nM T74312 CY8U1Q 57396557 IC50 = 7 nM T74312 CW4KG3 57396858 IC50 = 28 nM T74312 CE4FA1 57396924 IC50 = 350 nM T74312 CVQK90 57397197 IC50 = 10500 nM T74312 C1UZP2 57397437 IC50 = 95 nM T74312 C4J6UZ 57397845 IC50 < 1000 nM T74312 CWV96N 57398329 IC50 = 3 nM T74312 C8K1WJ 57398330 IC50 = 2 nM T74312 C59OYH 57398540 IC50 > 10000 nM T74312 CODG52 57398624 IC50 = 314 nM T74312 C3CEV7 57398898 IC50 = 6600 nM T74312 CM81VI 57398899 IC50 = 12400 nM T74312 CELC82 57398900 IC50 = 6200 nM T74312 CI76LU 57399379 IC50 = 6300 nM T74312 CBK02S 57399984 IC50 = 5 nM T74312 CNU4I7 57399985 IC50 = 5 nM T74312 CD9KF3 57399986 IC50 = 40 nM T74312 C4CW2G 57400284 IC50 > 1000 nM T74312 CM24WI 57400854 EC50 = 5300 nM T74312 CJ4YR1 57400855 IC50 = 44 nM T74312 C0BA7P 57401686 IC50 = 20 nM T74312 CH56JP 57401785 IC50 = 10 nM T74312 C7YMG1 57401804 IC50 > 1000 nM T74312 C20ZAX 57401805 IC50 = 10 nM T74312 C15YQW 57401806 IC50 = 20 nM T74312 CY5TJ9 57401807 IC50 = 5 nM T74312 C4L0SA 57401808 IC50 = 4 nM T74312 CE12CQ 57402393 IC50 = 4800 nM T74312 CQ3A5B 57402394 IC50 = 3100 nM T74312 C4J0OD 57403506 IC50 = 2 nM T74312 CN0M3Z 57403518 IC50 > 1000 nM T74312 CA71NH 57403845 IC50 > 1000 nM T74312 CZSM95 57412684 IC50 = 10 nM T74312 CXH6F3 57412768 IC50 = 6 nM T74312 C8R4FE 57991377 IC50 = 139.7 nM T74312 CD6ZP3 58009815 IC50 = 1800 nM T74312 CWU1Y3 58009825 IC50 = 440 nM T74312 C8S6MY 58010054 IC50 = 220 nM T74312 CM1B4V 58010265 IC50 = 240 nM T74312 CVK0G4 58056356 IC50 = 56 nM T74312 CH7L5N 58172700 IC50 = 882 nM T74312 CJ25EB 58299570 IC50 = 46 nM T74312 CJ4B6P 58299601 IC50 = 5 nM T74312 CU24DE 58299617 IC50 = 2 nM T74312 CDTZ75 58299762 IC50 = 17 nM T74312 CT78UE 58299836 IC50 = 11 nM T74312 CH1VI8 58299868 IC50 = 2 nM T74312 C1I0OB 58299870 IC50 = 17 nM T74312 CD87NL 58300031 IC50 = 43 nM T74312 C5RB1P 58300060 IC50 = 95 nM T74312 C63AEW 58300068 IC50 = 22 nM T74312 C1BJ9K 58300077 IC50 = 5 nM T74312 CT0U1H 58486131 IC50 = 1200 nM T74312 C4Y6PF 58486151 IC50 = 98 nM T74312 CCF5Y4 58486156 IC50 = 200 nM T74312 C2I3QW 58486157 IC50 = 97 nM T74312 C7ZKF5 58486186 IC50 = 45 nM T74312 CBF7L4 58486208 IC50 = 230 nM T74312 CM91GS 58486210 IC50 = 77 nM T74312 CQPU86 58486223 IC50 = 62 nM T74312 CB0Z6T 58486228 IC50 = 200 nM T74312 C3ZKB1 58486287 IC50 = 240 nM T74312 C51FBH 58486335 IC50 = 6500 nM T74312 C35FWX 58486367 IC50 = 3200 nM T74312 CB42EF 58557147 IC50 > 50000 nM T74312 C6BPR2 58985201 IC50 > 30000 nM T74312 C3L4JY 59176329 IC50 = 3 nM T74312 CXJ63M 59603829 IC50 < 10 nM T74312 CQEU96 59603842 IC50 = 1.9 nM T74312 COH62U 60097413 IC50 > 5000 nM T74312 C3JE8D 60142953 IC50 = 2 nM T74312 C6XA7U 60142955 IC50 = 4 nM T74312 CL0N9F 60143086 IC50 = 34 nM T74312 CZT65A 60143089 IC50 = 14 nM T74312 CSZA16 60155724 IC50 > 3600 nM T74312 C08VMZ 60198892 IC50 = 2 nM T74312 C4K8YJ 60198895 IC50 = 580 nM T74312 C5ZB2G 60199003 IC50 = 95 nM T74312 CN3W2C 60199004 IC50 = 72 nM T74312 CTR58Y 60199005 IC50 = 14 nM T74312 CFD0Q4 60202647 IC50 = 1 nM T74312 CHO3M7 66597981 IC50 = 157 nM T74312 C7W2XF 66597997 IC50 = 125 nM T74312 C52HRW 66598095 IC50 = 53 nM T74312 C5D3TJ 66598153 IC50 = 271 nM T74312 C51XCV 66781377 IC50 = 4 nM T74312 CV63UL 67240318 IC50 > 5000 nM T74312 C6D3QJ 67448476 IC50 = 44 nM T74312 C65XEF 67955686 IC50 = 320 nM T74312 CR7DN8 68032650 IC50 = 150 nM T74312 CS5C0R 68212798 IC50 = 3 nM T74312 C8I7GC 68293638 IC50 = 9100 nM T74312 C0HA8V 68783839 IC50 = 1 nM T74312 C5DGR9 69036886 IC50 = 8 nM T74312 CCS20X 69063773 IC50 = 40 nM T74312 CV3OL2 69403720 IC50 = 191.4 nM T74312 CLHG12 69403875 IC50 = 46 nM T74312 CZ7O5B 69404079 IC50 = 587 nM T74312 CD72BH 69404442 IC50 = 846 nM T74312 C8NDU6 69404540 IC50 = 119 nM T74312 CZ32PM 69404608 IC50 = 2.495 nM T74312 CAOE64 69412987 IC50 = 10.15 nM T74312 CDP96Z 69788774 IC50 = 33 nM T74312 CECZ23 70654418 IC50 = 4 nM T74312 CG50UJ 70654476 IC50 = 13 nM T74312 C4BS5T 70654492 IC50 = 10 nM T74312 CKP9E6 70654499 IC50 = 12 nM T74312 CAI3J4 70654537 IC50 = 30 nM T74312 CEXK08 70654539 IC50 = 5 nM T74312 C5NDK0 70654558 IC50 = 9 nM T74312 C0AP6Q 70654571 IC50 = 20 nM T74312 CRVS29 70654613 IC50 = 40 nM T74312 COV46X 70654614 IC50 = 27 nM T74312 CPF8W3 70654623 IC50 = 19 nM T74312 CVL6N9 70654642 IC50 = 18 nM T74312 CP0O5A 70654694 IC50 = 17 nM T74312 C9QS6O 70654709 IC50 = 16 nM T74312 C4INO3 70654745 IC50 = 13 nM T74312 CC0S3D 70654753 IC50 = 35 nM T74312 C7F4DB 70654775 IC50 = 4 nM T74312 C4I8WO 70654805 IC50 = 40 nM T74312 C5LFG2 70654826 IC50 = 280 nM T74312 CA0UR2 70654830 IC50 = 8 nM T74312 CWE94C 70654840 IC50 = 43 nM T74312 C23AJO 70654866 IC50 = 94 nM T74312 CS6I4T 70654868 IC50 = 7 nM T74312 CGU2P6 70654923 IC50 = 140 nM T74312 C59APG 70654958 IC50 = 18 nM T74312 C2LTI3 70654979 IC50 = 35 nM T74312 C6EK1V 70654997 IC50 = 10 nM T74312 CJAI19 70655010 IC50 = 14 nM T74312 CX3V5C 70655056 IC50 = 7 nM T74312 C49KEL 70655062 IC50 = 15 nM T74312 CW8XC7 70655063 IC50 = 52 nM T74312 CUYK36 70655070 IC50 = 17 nM T74312 CNQ56Y 70657170 IC50 = 19 nM T74312 C2A4PE 70660513 IC50 = 6 nM T74312 CF92MK 70660523 IC50 = 390 nM T74312 C7QL4R 70660524 IC50 = 21 nM T74312 C5U0EL 70661438 IC50 = 21 nM T74312 C98FWB 70661441 IC50 = 9 nM T74312 C03CKB 70661448 IC50 = 6 nM T74312 CEB12M 70681395 IC50 > 1000 nM T74312 CH27DE 70681409 IC50 > 1000 nM T74312 CN29RI 70681410 IC50 > 1000 nM T74312 CG93IE 70683519 IC50 > 900 nM T74312 CXSN14 70685622 IC50 > 1000 nM T74312 CL24MP 70687766 IC50 = 500 nM T74312 C4BLJ8 70688051 IC50 = 0.6 nM T74312 C51DHN 70689791 IC50 > 800 nM T74312 C6ITV3 70689792 IC50 = 200 nM T74312 CMLY63 70689816 IC50 = 300 nM T74312 C08ASR 70689830 IC50 > 1000 nM T74312 CGA43T 70690710 IC50 = 17 nM T74312 C4TF3G 70691955 IC50 > 1000 nM T74312 CTWD94 70691956 IC50 > 1000 nM T74312 CIK5N2 70691957 IC50 = 30 nM T74312 C8RZP3 70691958 IC50 = 300 nM T74312 C0XRC9 70691981 IC50 = 3000 nM T74312 C9RT8C 70693982 IC50 = 700 nM T74312 C2X1KJ 70694006 IC50 = 80 nM T74312 C54VLD 70694007 IC50 = 60 nM T74312 C6O3SM 70696108 IC50 = 200 nM T74312 CJH41B 70850449 IC50 = 480 nM T74312 C0JTH8 71166789 IC50 = 3286 nM T74312 C7SX3I 71450567 IC50 = 29 nM T74312 CYBE17 71452399 IC50 = 4.1 nM T74312 C2EI0Q 71452401 IC50 = 17 nM T74312 CKT60L 71455860 Ki = 494 nM T74312 CRQ6N1 71463084 IC50 = 14 nM T74312 CQY31T 71498139 IC50 = 8.5 nM T74312 C01XHF 71510730 IC50 = 218 nM T74312 C09YSR 71510731 IC50 = 288 nM T74312 C9DIK2 71512060 IC50 = 6810 nM T74312 C6HF8S 71521082 IC50 = 973.9 nM T74312 C9Z3AI 71521083 IC50 = 117.8 nM T74312 CCN01X 71547862 IC50 > 10000 nM T74312 CH62VU 71575112 IC50 = 1650 nM T74312 CX9I0D 71575113 IC50 = 1240 nM T74312 C7LG4R 71575114 IC50 = 1690 nM T74312 C5A8DG 71575115 IC50 = 260 nM T74312 C73JDI 71575116 IC50 = 2050 nM T74312 CV9UR5 71575210 IC50 = 20 nM T74312 C95HKC 71575211 IC50 = 83 nM T74312 COYB15 71575212 IC50 = 37 nM T74312 C29ZRL 71575213 IC50 = 5 nM T74312 C0H9JS 71575214 IC50 = 1590 nM T74312 CYNE63 71575215 IC50 = 79 nM T74312 C58JCR 71575322 IC50 = 4530 nM T74312 CG5T8U 71575323 IC50 = 7820 nM T74312 C3CO2D 71575324 IC50 > 10000 nM T74312 CUQ5M2 71575325 IC50 > 10000 nM T74312 CH2OJ3 71575326 IC50 = 7070 nM T74312 CR3U0E 71575327 IC50 > 10000 nM T74312 CJ8W6V 71575436 IC50 > 10000 nM T74312 C94WCB 71575437 IC50 > 10000 nM T74312 CDEF29 71575438 IC50 = 320 nM T74312 C6O3YU 71575541 IC50 = 96 nM T74312 C6AF9R 71575542 IC50 = 90 nM T74312 C12IXZ 71575543 IC50 = 4 nM T74312 CC23TP 71575544 IC50 = 11 nM T74312 C59CFR 71575545 IC50 = 59 nM T74312 CE06GM 71575546 IC50 = 54 nM T74312 CR4UT6 71575640 IC50 = 17 nM T74312 CRLI36 71575641 IC50 = 18 nM T74312 CRX81Q 71575642 IC50 = 3 nM T74312 CB6LS5 71658742 IC50 = 52 nM T74312 CIN8Q2 71658743 IC50 = 70 nM T74312 CEY10J 71658863 IC50 = 74 nM T74312 CC40FI 71658864 IC50 = 50 nM T74312 CN7TP5 71659100 IC50 = 22 nM T74312 C3AMG7 71659101 IC50 = 66 nM T74312 CD84KP 71659102 IC50 = 16 nM T74312 CS3Q2M 71659227 IC50 = 17 nM T74312 CYSZ68 71659355 IC50 = 26 nM T74312 C1FAU8 71679855 IC50 = 380 nM T74312 C9ID4J 71716376 IC50 = 363 nM T74312 CL8JN9 71718823 IC50 = 1074 nM T74312 C63RGU 71718904 IC50 > 10000 nM T74312 CKM7P3 71720012 IC50 = 449 nM T74312 CDN3T2 71720643 IC50 = 1371 nM T74312 C60BIX 71763463 IC50 = 100 nM T74312 CKZ5W3 71815103 IC50 = 16.2 nM T74312 CCV20F 71815104 IC50 = 106 nM T74312 C4Q6FE 71815105 IC50 = 11 nM T74312 CJ9OX6 71815106 IC50 = 16.6 nM T74312 C2R4SM 71815390 IC50 = 8.6 nM T74312 CP8UA4 71815638 IC50 = 201.1 nM T74312 C1EHU9 71815639 IC50 = 58.2 nM T74312 CSA3K0 71815640 IC50 = 333.9 nM T74312 CGV20M 71815692 IC50 > 1000 nM T74312 C8X3RA 71815744 IC50 > 1000 nM T74312 CUQK27 71815745 IC50 > 1000 nM T74312 C38MPZ 71815746 IC50 = 31.7 nM T74312 C3Z9XP 71815811 IC50 = 675.8 nM T74312 COP37R 71815812 IC50 > 1000 nM T74312 CZHF40 71815813 IC50 > 1000 nM T74312 CUP32D 71815814 IC50 = 384.8 nM T74312 CAU21X 71815815 IC50 > 1000 nM T74312 CC1Q2L 71815881 IC50 > 1000 nM T74312 C6NV5E 71815882 IC50 > 1000 nM T74312 CC1T4S 71815884 IC50 = 133.5 nM T74312 CWOS79 71815948 IC50 = 2.7 nM T74312 CO6EQ1 71815949 IC50 > 1000 nM T74312 CBF15Z 71816016 IC50 = 405.5 nM T74312 C3ZX5P 71816017 IC50 = 111.1 nM T74312 CG01VI 71816018 IC50 > 1000 nM T74312 CCM0E5 71816019 IC50 = 16.3 nM T74312 CWUH04 71816084 IC50 = 57.1 nM T74312 CY8CM3 71816085 IC50 = 79.5 nM T74312 C3VT2G 71816086 IC50 > 1000 nM T74312 CD28XR 71816087 IC50 = 0.5 nM T74312 CPU41Q 71816088 IC50 = 4.4 nM T74312 CSA2J6 72187684 IC50 = 312 nM T74312 CB64IQ 72194525 IC50 = 0.438 nM T74312 CRFP28 72194526 IC50 = 0.623 nM T74312 C96VXT 72194909 IC50 = 2.56 nM T74312 CH0XR4 72195175 IC50 = 0.27 nM T74312 C9P6NG 72195176 IC50 = 2.06 nM T74312 C97DTU 72195318 IC50 = 0.47 nM T74312 C2K3DV 72195319 IC50 = 6.15 nM T74312 CY9M6J 72195452 IC50 = 3.52 nM T74312 C0DZ9T 72195453 IC50 = 0.576 nM T74312 C94SKQ 72195454 IC50 = 0.384 nM T74312 CUZV18 72195456 IC50 = 1.37 nM T74312 CSM37G 72195457 IC50 = 0.167 nM T74312 C4N9OI 72202732 IC50 = 1317 nM T74312 C7FJB9 72202734 IC50 = 1869 nM T74312 CSW20D 72202735 IC50 = 5449 nM T74312 CV23JN 72202867 IC50 = 1528 nM T74312 CW8HV3 72202868 IC50 = 1056 nM T74312 C6FZA2 72202870 IC50 = 3589 nM T74312 C8WC6P 72202999 IC50 = 2920 nM T74312 CA7Y5H 72203000 IC50 = 165 nM T74312 CW18BO 72203003 IC50 = 1136 nM T74312 CI63WE 72203004 IC50 = 47 nM T74312 C0K6SQ 72203136 IC50 = 4413 nM T74312 C5BP6D 72712977 IC50 = 29 nM T74312 CUS2R1 72712978 IC50 = 34 nM T74312 C5ZU4Y 72713172 IC50 = 108 nM T74312 CUDS15 72713174 IC50 = 184 nM T74312 CH93FM 72713175 IC50 = 384 nM T74312 CH3K0R 72713176 IC50 = 173 nM T74312 C9LA5P 72713177 IC50 = 1747 nM T74312 CK3N8G 72713385 IC50 = 153 nM T74312 CA58QS 72734886 IC50 = 162 nM T74312 C8SIL6 73349435 IC50 = 1.08 nM T74312 C7F0YR 73353451 IC50 = 26 nM T74312 CZN1Y6 73354960 IC50 = 20 nM T74312 C1V3NZ 73425588 IC50 = 14 nM T74312 C2PAK9 73438493 IC50 = 20 nM T74312 C4U5NV 73442760 IC50 = 18000 nM T74312 CGDB30 74538658 IC50 = 50 nM T74312 CQ4ZH2 74538669 IC50 = 320 nM T74312 CBAT06 76071144 IC50 = 20 nM T74312 C29EZO 76871930 IC50 = 500 nM T74312 C9MPZ1 77107163 IC50 = 4 nM T74312 CNH79R 77107360 IC50 = 5 nM T74312 CZ97VP 86294733 IC50 = 20 nM T74312 CB5NJ4 86302541 IC50 > 10000 nM T74312 CPG3A5 86302574 IC50 > 30000 nM T74312 C08WGI 86566799 IC50 = 8.78 nM T74312 CIV48L 86760649 IC50 = 113 nM T74312 CUNA57 88876306 IC50 = 20 nM T74312 CDW95X 88876318 IC50 = 10 nM T74312 CE6RY9 88876331 IC50 = 73 nM T74312 CT1L6U 88876351 IC50 = 320 nM T74312 C31EBZ 88876355 IC50 = 38 nM T74312 CVEA94 88876366 IC50 = 33 nM T74312 CHIZ70 89495685 IC50 = 1 nM T74312 CS6IA4 89495748 IC50 = 3 nM T74312 CW1OS0 89495775 IC50 = 1.2 nM T74312 C1HW4B 89735655 IC50 = 580 nM T74312 C61TVX 89857999 IC50 > 1000 nM T74312 CQW14S 89858004 IC50 = 908.9 nM T74312 CA4F0J 89858007 IC50 = 10 nM T74312 CF17VX 89858058 IC50 = 41.4 nM T74312 C2ECL1 89858082 IC50 = 179.8 nM T74312 CQ2OB9 90292687 IC50 = 238 nM T74312 CHI39S 90292823 IC50 = 709 nM T74312 C4EFG8 90479851 IC50 = 1070 nM T74312 CK6V9J 90644118 IC50 = 673 nM T74312 C5S3YB 90645165 IC50 = 9.28 nM T74312 CY0UC4 90645194 IC50 > 10000 nM T74312 C9AJE8 90647152 IC50 = 790 nM T74312 C19UKQ 90654460 IC50 = 3 nM T74312 C9Y7JE 90654461 IC50 = 0.3 nM T74312 C5RV8E 90654462 IC50 = 6 nM T74312 CILZ92 90654463 IC50 = 1 nM T74312 C19AQS 90654464 IC50 = 2 nM T74312 CMSI40 90654465 IC50 = 0.6 nM T74312 CUT04P 90654466 IC50 = 0.2 nM T74312 CE8AI2 90654467 IC50 = 6 nM T74312 C1LN6H 90654468 IC50 = 8 nM T74312 CPZM73 90654469 IC50 = 8 nM T74312 CBT0X9 90654470 IC50 = 3 nM T74312 C9CM8Y 90654471 IC50 = 0.6 nM T74312 CJK82D 90667370 IC50 = 1300 nM T74312 C3K8QL 90682433 IC50 = 9.28 nM T74312 CJQ5N6 91936970 IC50 = 322000 nM T74312 CAU45T 91971978 IC50 > 30000 nM T74312 C64SIO 92042864 IC50 = 13 nM T74312 C8F7XO 92131166 IC50 = 8.91 nM T74312 CGEQ73 92135951 IC50 = 5 nM T74312 CK72FW 102129497 IC50 = 3.49 nM T74312 CZ4E1B 110856540 IC50 > 2000 nM T74312 C64MRE 110861543 IC50 > 2000 nM T74312 C8WS5U 110861626 IC50 > 2000 nM T74312 C0LCN1 118105340 IC50 = 28 nM T74312 CL2DH6 118433464 IC50 = 61 nM T74312 C01OAD 118433470 IC50 = 316 nM T74312 C9ENZ0 118433703 IC50 = 3.4 nM T74312 CQU1R4 118443520 IC50 = 543 nM T74312 C8OSQ4 118443521 IC50 = 109 nM T74312 CAM76F 118443524 IC50 = 544 nM T74312 C3DEP2 118443546 IC50 = 66 nM T74312 CGO6B1 118443548 IC50 = 8299 nM T74312 CADG96 118443549 IC50 = 37 nM T74312 CM92EG 118443553 IC50 = 202 nM T74312 CVWR20 118443556 IC50 = 4372 nM T74312 CC9FK0 118443560 IC50 = 162 nM T74312 CRZ68N 118443583 IC50 = 49 nM T74312 C9I5MC 118443585 IC50 = 107 nM T74312 CE42TF 118443586 IC50 = 1296 nM T74312 C5YJT1 118443594 IC50 = 19 nM T74312 CL0YO5 118443595 IC50 = 2.5 nM T74312 CG3K5V 118443597 IC50 = 189 nM T74312 C12WAU 118446433 IC50 = 214 nM T74312 CFBY13 118446434 IC50 = 1.5 nM T74312 CK92PQ 118464648 IC50 = 54.37 nM T74312 CZ6YL3 118464657 IC50 = 521 nM T74312 CSM56H 118464669 IC50 = 11.38 nM T74312 CK6M1N 118464670 IC50 = 74.97 nM T74312 C8H9BY 118489441 IC50 = 50 nM T74312 C3H2EM 118489443 IC50 = 82 nM T74312 C8SL5D 118489445 IC50 = 11 nM T74312 CXLI69 118489448 IC50 = 36 nM T74312 CHY69E 118489449 IC50 = 38 nM T74312 CZBF45 118489450 IC50 = 28 nM T74312 C7COI2 118489453 IC50 = 6 nM T74312 CRA1T5 118489454 IC50 = 56 nM T74312 CR0N4P 118489455 IC50 = 657 nM T74312 CQA1O7 118489457 IC50 = 52 nM T74312 CN3O6F 118489458 IC50 = 8 nM T74312 CYZD10 118489459 IC50 = 42 nM T74312 C59USA 118489460 IC50 = 62 nM T74312 CI51DY 118489464 IC50 = 2 nM T74312 CKT91A 118489466 IC50 = 66 nM T74312 CK1UO8 118489472 IC50 = 73 nM T74312 C6QI9N 118489473 IC50 = 53 nM T74312 CM3Q1P 118489479 IC50 = 294 nM T74312 CBQ7H6 118489480 IC50 = 8 nM T74312 CU2O3L 118489481 IC50 = 10 nM T74312 C19LOD 118489482 IC50 = 27 nM T74312 COM84Z 118491814 IC50 = 217 nM T74312 CKS7R3 118491815 IC50 = 80 nM T74312 C82PEL 118491816 IC50 = 449 nM T74312 CDK5G4 118687517 IC50 = 18.6 nM T74312 CY7BI2 118706214 IC50 > 10000 nM T74312 C2IN3C 118710236 IC50 = 6.4 nM T74312 CF2YR1 118710237 IC50 = 2.1 nM T74312 C4AHL2 118711367 IC50 = 1000 nM T74312 CH6D8R 118713361 IC50 > 1000 nM T74312 C7DH4V 118713364 IC50 > 1000 nM T74312 CWO9B7 118715995 IC50 = 390 nM T74312 CV37AU 118722005 IC50 >= 30000 nM T74312 CJ2GP0 118722006 IC50 = 8310 nM T74312 CCPX67 118722007 IC50 = 9610 nM T74312 C1BTE4 118722008 IC50 = 10520 nM T74312 C7OG6R 118722009 IC50 = 15900 nM T74312 C3TO7Q 118722010 IC50 = 1110 nM T74312 CI76QW 118722011 IC50 = 2250 nM T74312 C4EPD2 118722012 IC50 = 4230 nM T74312 CRP21J 118722013 IC50 >= 30000 nM T74312 CQY3R9 118722014 IC50 >= 30000 nM T74312 CSM2K7 118722015 IC50 >= 30000 nM T74312 C01WPE 118722016 IC50 >= 30000 nM T74312 CN26HZ 118722017 IC50 = 3370 nM T74312 CR4GQ6 118722018 IC50 = 1340 nM T74312 C7X4WF 118722019 IC50 = 3030 nM T74312 CL2NC0 118722020 IC50 = 150 nM T74312 C4WI3S 118722021 IC50 = 8870 nM T74312 C67NJM 118722022 IC50 = 1740 nM T74312 C8JF6I 118722023 IC50 = 1640 nM T74312 CU1BZ9 118722024 IC50 = 2100 nM T74312 CQ6M4O 118722025 IC50 = 3010 nM T74312 CU2C4J 118722026 IC50 = 14150 nM T74312 C0ER7J 118722027 IC50 >= 30000 nM T74312 CPN16I 118722028 IC50 >= 30000 nM T74312 CAQ6F2 118722029 IC50 >= 30000 nM T74312 C90DEI 118722030 IC50 >= 30000 nM T74312 C3KLI5 118723185 IC50 = 36000 nM T74312 C9XNG5 118724918 IC50 > 1000 nM T74312 CHT6K9 118728811 Ki > 4000 nM T74312 CUA3Y2 118728812 Ki = 1100 nM T74312 CDQ78G 118728813 Ki > 4000 nM T74312 CZ6XL7 118728814 Ki = 210 nM T74312 CMO67K 118728815 Ki = 800 nM T74312 CR2M0Q 118728816 Ki = 2800 nM T74312 C62SCL 118728817 Ki > 4000 nM T74312 CSB30C 118728819 Ki = 1200 nM T74312 CV7XU8 118728820 Ki = 160 nM T74312 C3J1EX 118728821 Ki = 4000 nM T74312 CIWB78 118728822 Ki = 1400 nM T74312 CP18SE 118728823 Ki = 150 nM T74312 CM42CA 118728824 Ki = 970 nM T74312 C9Q7CL 118728825 Ki = 1800 nM T74312 CCR3S0 118728826 Ki = 840 nM T74312 C2UTG0 118733889 IC50 = 51 nM T74312 CQ40WL 118733891 IC50 = 15 nM T74312 CAK5L1 118733892 IC50 = 470 nM T74312 C5X4ZV 118733893 IC50 = 190 nM T74312 C82IGC 118733894 IC50 = 160 nM T74312 CT0CY7 118733895 IC50 = 41 nM T74312 CV72AB 118733896 IC50 = 230 nM T74312 CEXY06 118733897 IC50 = 550 nM T74312 COP6V0 118733898 IC50 = 300 nM T74312 CWK4J7 118733899 IC50 = 16 nM T74312 CJ7PF4 118733901 IC50 = 430 nM T74312 C12VBU 118733902 IC50 = 440 nM T74312 CNL96I 118733903 IC50 = 78 nM T74312 CN2SA5 118734641 IC50 = 180 nM T74312 CF6J5Q 118734642 IC50 = 108 nM T74312 CMHF86 118734643 IC50 = 87 nM T74312 CUE83V 118734644 IC50 = 556 nM T74312 C67IDL 118734645 IC50 = 1256 nM T74312 C26ZJS 118734647 IC50 = 217 nM T74312 CM5A9U 118734648 IC50 = 221 nM T74312 C7HP6N 118734649 IC50 = 833 nM T74312 CVIN49 118734650 IC50 = 272 nM T74312 CI1Q9W 118736571 IC50 = 1750 nM T74312 C75PHN 119058124 IC50 = 180 nM T74312 C9R4YK 121453018 IC50 > 12500 nM T74312 C2KJB6 121453019 IC50 = 1020 nM T74312 CQD35J 121453020 IC50 > 12500 nM T74312 CVUA52 121453021 IC50 = 70 nM T74312 CPO56W 121453023 IC50 = 1230 nM T74312 CGO2A7 121453024 IC50 = 10190 nM T74312 CYTA98 121453025 IC50 = 1670 nM T74312 C63FBC 121453027 IC50 = 3600 nM T74312 CDR37K 121453028 IC50 > 12500 nM T74312 CH7G2V 121453029 IC50 = 5950 nM T74312 CV7AP5 121453030 IC50 = 3080 nM T74312 CK7Y1O 121453031 IC50 = 12500 nM T74312 CETM30 121453032 IC50 = 2330 nM T74312 CZP58J 121453033 IC50 = 1510 nM T74312 C4G8LB 121453034 IC50 > 12500 nM T74312 C2C1YX 121453035 IC50 = 12500 nM T74312 C0PK8F 121453039 IC50 = 410 nM T74312 CB5L7Y 121453042 IC50 = 6320 nM T74312 C7D2AG 121453043 IC50 = 1030 nM T74312 CM54LG 121453044 IC50 = 340 nM T74312 CAJR21 121453047 IC50 > 12500 nM T74312 CN14PR 121453048 IC50 > 12500 nM T74312 CX1IH7 121453049 IC50 = 7020 nM T74312 CTZ31N 121453054 IC50 > 12500 nM T74312 CFZ7B1 121453055 IC50 = 120 nM T74312 CTQ84B 121453056 IC50 = 6860 nM T74312 CFCJ46 121453057 IC50 = 6000 nM T74312 C1N5JL 121453058 IC50 = 1910 nM T74312 CKE0Y6 121453061 IC50 = 1510 nM T74312 CO7W3M 121453062 IC50 = 2100 nM T74312 CFWC68 121453063 IC50 = 1850 nM T74312 CDP75O 121453065 IC50 = 2750 nM T74312 CW71GA 121453067 IC50 = 100 nM T74312 CF48BP 121453070 IC50 = 560 nM T74312 CT71XV 121453071 IC50 = 12500 nM T74312 C4P3UT 121453072 IC50 = 3550 nM T74312 CZM16W 121453073 IC50 = 2750 nM T74312 CBJ1R7 121453075 IC50 = 1290 nM T74312 CO06WT 121453076 IC50 = 2560 nM T74312 CP2E0L 121453077 IC50 > 12500 nM T74312 CUVF37 121453078 IC50 = 2940 nM T74312 C7VBJ5 121453079 IC50 = 2210 nM T74312 CE2LQ0 121453080 IC50 > 12500 nM T74312 CW64CM 121453081 IC50 = 200 nM T74312 C8GA4Q 121453082 IC50 = 190 nM T74312 CY9AI7 121453084 IC50 = 12500 nM T74312 CM0SH9 121453085 IC50 = 3600 nM T74312 C5BRD3 121453086 IC50 > 12500 nM T74312 CT5I9L 121453088 IC50 = 340 nM T74312 CW9G8N 121453089 IC50 > 12500 nM T74312 CHR63C 121453090 IC50 = 740 nM T74312 CPEO87 121453091 IC50 > 12500 nM T74312 CM9QC6 121453092 IC50 > 12500 nM T74312 C9FWC7 121453093 IC50 = 4300 nM T74312 CHC6E5 121453094 IC50 > 12500 nM T74312 CT17HO 121453095 IC50 > 12500 nM T74312 C5S7IF 121453097 IC50 = 2100 nM T74312 CR07AV 121453098 IC50 = 2200 nM T74312 CN09GO 121453099 IC50 = 3520 nM T74312 C1UX0R 121453100 IC50 > 12500 nM T74312 CQD7K0 121453101 IC50 = 1210 nM T74312 CX9ZN7 121453102 IC50 = 5990 nM T74312 CS3GN2 121453103 IC50 = 3590 nM T74312 CZ7QE6 121453104 IC50 > 12500 nM T74312 CSO0X1 121453105 IC50 = 6040 nM T74312 CS53XT 121453106 IC50 = 4950 nM T74312 CQ1Y4N 121453109 IC50 > 12500 nM T74312 C3BQ4I 121453110 IC50 = 2740 nM T74312 CY6G1L 121453113 IC50 = 5650 nM T74312 C0LN8D 121453114 IC50 > 12500 nM T74312 CE7K2C 121453115 IC50 = 7580 nM T74312 CK14UG 121453117 IC50 = 5690 nM T74312 C8C7SX 121453118 IC50 = 4850 nM T74312 CTA5X1 121453119 IC50 = 12500 nM T74312 CS04NG 121453120 IC50 = 3410 nM T74312 CBDH54 121453123 IC50 > 12500 nM T74312 CX25VE 121453125 IC50 = 190 nM T74312 C4UB2S 121453126 IC50 = 150 nM T74312 C7N3IL 121453127 IC50 = 9310 nM T74312 CS10RG 121453129 IC50 = 11370 nM T74312 CK32TJ 121453130 IC50 = 1510 nM T74312 CR3A0S 121453132 IC50 > 12500 nM T74312 CGYK87 121453133 IC50 = 2170 nM T74312 CCDK68 121453136 IC50 = 2260 nM T74312 CAUZ05 121453137 IC50 = 3220 nM T74312 C85XGM 121453138 IC50 = 6430 nM T74312 C5OP2I 121453139 IC50 > 12500 nM T74312 C78RAD 121453140 IC50 = 5010 nM T74312 C8JPO7 121453141 IC50 > 12500 nM T74312 CVO9E0 121453142 IC50 > 12500 nM T74312 C67OZV 121453143 IC50 = 3070 nM T74312 CKW5Z0 121453144 IC50 > 12500 nM T74312 C2W3KQ 121453145 IC50 = 80 nM T74312 C8TQ0F 121453146 IC50 > 12500 nM T74312 CTR7H8 121453147 IC50 = 1340 nM T74312 CS2EI7 121453148 IC50 = 2810 nM T74312 CIR0W2 121453149 IC50 = 4500 nM T74312 C3Z4IE 121453152 IC50 = 2530 nM T74312 C7A4PU 121453153 IC50 = 5620 nM T74312 CB5K6U 121453154 IC50 = 12500 nM T74312 CBZL42 121453155 IC50 = 30 nM T74312 C20AWX 121453157 IC50 = 810 nM T74312 C1TO4F 121453158 IC50 = 1770 nM T74312 CF8H4A 121453160 IC50 > 12500 nM T74312 CE8W7D 121453161 IC50 = 1160 nM T74312 C26AUC 121453162 IC50 = 9150 nM T74312 CJ2S4O 121453163 IC50 > 12500 nM T74312 CD8IK9 121453164 IC50 = 8660 nM T74312 CHS23V 121453167 IC50 = 2060 nM T74312 CGLM28 121459818 IC50 = 1350 nM T74312 CHN4K7 121459819 IC50 = 10630 nM T74312 C4B3UF 121459821 IC50 = 3800 nM T74312 CS0A6M 121459822 IC50 = 4190 nM T74312 C7QE2J 121513893 EC50 < 30 nM T74312 C08KEM 122179540 IC50 = 720 nM T74312 C3AJ4C 122179546 IC50 = 8100 nM T74312 CG0RP7 122179547 IC50 = 3300 nM T74312 C1A0SQ 122179548 IC50 = 4300 nM T74312 C42GSX 122180520 Ki > 4000 nM T74312 CN81HR 122181799 IC50 = 79 nM T74312 C2D8UA 122181800 IC50 = 49 nM T74312 CMU6G9 122181801 IC50 = 22 nM T74312 C8DJ3K 122181802 IC50 = 520 nM T74312 CR9FQ7 122181803 IC50 = 83 nM T74312 CTS2C6 122181804 IC50 = 850 nM T74312 CWA94G 122182409 IC50 = 134 nM T74312 C9MIL3 122188249 IC50 = 32 nM T74312 C53AYQ 122188250 IC50 = 4628 nM T74312 CZO41H 122188251 IC50 > 10000 nM T74312 CLW25J 122188252 IC50 = 154 nM T74312 C23PIE 122188253 IC50 > 10000 nM T74312 CE41KZ 122188254 IC50 > 10000 nM T74312 CHQT85 122188255 IC50 = 7791 nM T74312 CLAD59 122188256 IC50 = 90 nM T74312 CI0W3V 122188257 IC50 = 8855 nM T74312 C3BXR2 122188258 IC50 > 10000 nM T74312 C67GYV 122188259 IC50 = 3301 nM T74312 CE81FB 122188260 IC50 > 10000 nM T74312 CG8VX5 122188261 IC50 = 1913 nM T74312 C9ZKA1 122188262 IC50 = 8882 nM T74312 CQF9I2 122188263 IC50 = 5047 nM T74312 COGF57 122188264 IC50 > 10000 nM T74312 CV8D3O 122188265 IC50 = 6264 nM T74312 CPQ89G 122188266 IC50 = 33 nM T74312 CA4LH8 122188267 IC50 > 10000 nM T74312 CO9LT3 122188268 IC50 = 6456 nM T74312 CRH4E1 122188269 IC50 = 21 nM T74312 CXT3E9 122188270 IC50 = 97 nM T74312 CVEB28 122188271 IC50 = 0.762 nM T74312 C5E7WK 122188272 IC50 = 3.12 nM T74312 CWIR28 122188273 IC50 = 7.48 nM T74312 CB6I5A 122188274 IC50 > 10 nM T74312 CA8VH1 122188275 IC50 = 0.212 nM T74312 C1XAP9 122188276 IC50 = 1.19 nM T74312 C0BLT6 122188277 IC50 > 10 nM T74312 CA6V5M 122188278 IC50 = 15.1 nM T74312 CP9H3I 122188279 IC50 = 0.166 nM T74312 CV89ZC 122188280 IC50 = 0.374 nM T74312 C2D5TF 122188281 IC50 = 0.177 nM T74312 C93VST 122188282 IC50 = 1.9 nM T74312 C5FGI7 122188283 IC50 = 1.28 nM T74312 CJY4C1 122188365 IC50 = 0.123 nM T74312 CM8X3C 122192463 IC50 = 22 nM T74312 C4Q7DT 122192464 IC50 = 95 nM T74312 C4X7SD 122192466 IC50 = 22 nM T74312 CJ6RO8 122193596 IC50 > 10000 nM T74312 C0T6VF 123561371 IC50 > 10000 nM T74312 C7G6IA 123944769 IC50 = 6320 nM T74312 CDL2V4 124005596 IC50 = 3970 nM T74312 CBYC49 126617676 IC50 < 10 nM T74312 C8KXV1 127025843 IC50 > 1000 nM T74312 CKWM43 127026646 IC50 = 110 nM T74312 C83LME 127026647 IC50 = 61 nM T74312 C7FPS1 127026648 IC50 = 95 nM T74312 CCH34N 127026649 IC50 = 90 nM T74312 CYG42Z 127026951 IC50 = 43 nM T74312 C5I3EH 127028830 IC50 = 46 nM T74312 CU4F8X 127028831 IC50 = 42 nM T74312 CZVW52 127028832 IC50 = 23 nM T74312 CDS6B4 127028833 IC50 = 56 nM T74312 C3E7FZ 127028834 IC50 = 9 nM T74312 CX13PS 127029131 IC50 > 2000 nM T74312 C1XD6R 127029809 IC50 = 2.15 nM T74312 CI1E5W 127029864 IC50 = 2.06 nM T74312 CTVL57 127031501 IC50 = 107 nM T74312 CKS28E 127034802 IC50 = 85.7 nM T74312 CKX40V 127037812 IC50 > 10000 nM T74312 C70RUP 127038480 IC50 > 10000 nM T74312 C3WCN8 127041777 IC50 > 10000 nM T74312 CC1VO7 127047444 IC50 = 280 nM T74312 CB6EI5 127048964 IC50 = 946 nM T74312 C72QDX 127049934 IC50 = 5707 nM T74312 C6WAN3 127050277 IC50 = 356 nM T74312 C3A7ZV 127050278 IC50 = 34 nM T74312 CSC97B 127050279 IC50 = 1526 nM T74312 C40TXA 127050280 IC50 = 6 nM T74312 CG1H7C 127051183 IC50 = 424 nM T74312 CQC30S 127051184 IC50 = 31 nM T74312 CSP90J 127051185 IC50 = 143 nM T74312 C19QLG 127051473 IC50 = 114 nM T74312 C5GQ4L 127051474 IC50 = 280 nM T74312 CU5QJ9 127051475 IC50 = 1577 nM T74312 CY2CW9 127051476 IC50 = 692 nM T74312 C62RLP 127051768 IC50 = 126 nM T74312 C3ORU9 127052113 IC50 = 4 nM T74312 C6RBC4 127052114 IC50 = 96 nM T74312 CZK3D8 127052115 IC50 = 40 nM T74312 C8QKM6 127052116 IC50 = 62 nM T74312 C1DM7O 127052427 IC50 = 83 nM T74312 CQ50XO 127052428 IC50 = 14 nM T74312 CWS5C4 129245211 IC50 = 30 nM T74312 CH91ON 129245363 IC50 = 114 nM T74312 CA2N5C 129245517 IC50 = 17 nM T74312 C0E2RU 129245526 IC50 = 37 nM T74312 C52PNC 129245623 IC50 = 0.3 nM T74312 CEYK58 129245795 IC50 = 9 nM T74312 COR37Y 129245842 IC50 = 173 nM T74312 CKB5C8 129245918 IC50 = 69 nM T74312 CQJK71 129246093 IC50 = 10 nM T74312 C0GC7N 129246130 IC50 = 11 nM T74312 CCF8W2 129261617 IC50 = 6 nM T74312 CG5O2J 129261641 IC50 = 9 nM T74312 C6NQG3 131704413 IC50 = 14 nM T74312 C0AV5D 131801161 IC50 = 0.54 nM T74312 CUO0C5 132156633 IC50 > 10000 nM T74312 C6OMB1 132204257 EC50 < 10 nM T74312 CJ04HZ 132585195 IC50 = 2 nM T74312 C8I7HV 132602209 IC50 = 5 nM T74312 CI2YE9 132606873 IC50 = 188 nM T74312 C53OJM 132607333 IC50 = 268.81 nM T74312 CR3C9O 132819862 IC50 = 0.63 nM T74312 CMI3Q0 132819888 IC50 = 400 nM T74312 CM06HV 133081975 IC50 = 8 nM T74312 C0TA9U 134132267 IC50 < 340 nM T74312 C7JC5K 134132904 IC50 = 7.5 nM T74312 C5DSV1 134134351 IC50 = 63 nM T74312 CYB46P 134135659 IC50 = 370 nM T74312 CDH31O 134136945 IC50 = 12 nM T74312 C46XTD 134138113 IC50 = 250 nM T74312 CK75ZI 134138785 IC50 = 56 nM T74312 CCE1O4 134138988 IC50 = 6.8 nM T74312 C9V4CG 134140406 IC50 = 29 nM T74312 CXRQ96 134140562 IC50 = 9.478 nM T74312 C5C4TS 134141052 IC50 = 1000 nM T74312 CWI41J 134141468 IC50 = 84 nM T74312 CYM06R 134142159 IC50 = 470 nM T74312 CZB68J 134142873 IC50 = 26 nM T74312 CX03CP 134143856 IC50 = 280 nM T74312 C5C2TA 134144975 IC50 = 12 nM T74312 CDO52G 134145027 IC50 = 3.769 nM T74312 CE12IN 134145489 IC50 = 550 nM T74312 CT5Y1Q 134146356 IC50 = 6.427 nM T74312 CM4U6L 134147181 IC50 = 8.9 nM T74312 CBES34 134147807 IC50 = 12 nM T74312 CUKE45 134147919 IC50 = 8.19 nM T74312 C60FLZ 134148014 IC50 = 9.6 nM T74312 CDUX09 134148124 IC50 = 160 nM T74312 CRLD28 134148597 IC50 = 0.334 nM T74312 CGIT02 134149104 IC50 = 6.3 nM T74312 C4CA2M 134149641 IC50 = 100 nM T74312 C36GLZ 134150279 IC50 = 2.5 nM T74312 CZ42MI 134150952 IC50 = 32 nM T74312 C39AMZ 134151100 IC50 = 8.1 nM T74312 C10BFN 134151512 IC50 = 70 nM T74312 C8M3RH 134152780 IC50 = 5.4 nM T74312 C5PV8R 134153049 IC50 = 20 nM T74312 CG9C3K 134153486 IC50 = 27.2 nM T74312 C4M7XF 134153576 IC50 = 37 nM T74312 C4AR9L 134153778 IC50 = 68 nM T74312 C6GC3U 134154700 IC50 = 130 nM T74312 CL7FG6 134155241 IC50 = 16.78 nM T74312 C20PJY 134156194 IC50 = 13 nM T74312 CHN5R6 134156911 IC50 = 75 nM T74312 C70ZRI 134157187 IC50 = 13 nM T74312 CIK38Q 134229735 IC50 = 27.9 nM T74312 C2AN7T 134611886 IC50 > 100000 nM T74312 CLCO61 135398510 IC50 = 1 nM T74312 CX8ID4 135418376 IC50 > 10000 nM T74312 C3A1LH 135422898 IC50 = 209 nM T74312 CR2F3P 135443448 IC50 = 280 nM T74312 C8GZ2B 135449326 Ki = 750 nM T74312 CPZH64 135468069 IC50 > 10000 nM T74312 CKD6H2 135481175 IC50 = 62 nM T74312 COBA59 135482273 IC50 = 359 nM T74312 CZO92B 135505769 IC50 = 82 nM T74312 CTB7R2 135564980 IC50 = 2 nM T74312 CI47VJ 135566923 IC50 = 20 nM T74312 CPHG43 135567142 IC50 = 5 nM T74312 CG2LO6 135567179 IC50 = 5.4 nM T74312 CAX7S0 135567181 IC50 = 35000 nM T74312 CPV59N 135685787 Ki = 130 nM T74312 CN5PS2 135800260 IC50 < 10000 nM T74312 C01HMT 135932346 IC50 = 35 nM T74312 CF1PS8 135934877 Ki = 66 nM T74312 CTRL59 135976660 Ki = 290 nM T74312 CYXR26 135985503 IC50 = 17 nM T74312 C4RL7Q 135985508 IC50 = 180 nM T74312 C3M7EP 135985511 IC50 = 49 nM T74312 CA46HS 135988914 IC50 = 50 nM T74312 CJE79B 135988932 IC50 = 120 nM T74312 C86BZJ 135988997 IC50 = 35 nM T74312 C5BDV8 135989018 IC50 = 72 nM T74312 CD7L3X 135989019 IC50 = 27 nM T74312 CJID74 136013449 IC50 = 27300 nM T74312 CHA4N2 136013680 IC50 > 10 nM T74312 C3YL4I 136042193 IC50 = 39 nM T74312 C1PCJ3 136042251 IC50 = 7300 nM T74312 CJ7U4C 136053657 IC50 = 366.7 nM T74312 CG1R7B 136087060 IC50 = 2300 nM T74312 CS4R2M 136098630 IC50 = 4 nM T74312 CWM2S3 136098631 IC50 = 111 nM T74312 CI9C0K 136108929 IC50 > 10000 nM T74312 CQ84IZ 136180335 Ki > 4000 nM T74312 CZ7EX0 136183413 IC50 = 60 nM T74312 CC52HL 136189674 IC50 > 3600 nM T74312 CDT7E4 136211077 IC50 > 100 nM T74312 C9RE8D 136215817 IC50 = 496.3 nM T74312 C1YUD0 136219394 IC50 > 10 nM T74312 CAY7U9 136236280 IC50 = 47 nM T74312 CRV68G 136254210 IC50 = 35 nM T74312 CIU8W3 136254389 IC50 > 10 nM T74312 CFQO70 136375226 IC50 = 28 nM T74312 CC8Q2D 136375233 IC50 = 140 nM T74312 C5PZ9U 137355929 IC50 = 24 nM T74312 C3Z7BX 137355931 IC50 = 0.1 nM T74312 CPF20O 137355933 IC50 > 1000 nM T74312 C37GOF 137355935 IC50 = 63 nM T74312 C9PVK0 137355939 IC50 = 35 nM T74312 C01WQT 137355941 IC50 = 163 nM T74312 CV9MO4 137355952 IC50 = 43 nM T74312 CWPA09 137355957 IC50 = 35 nM T74312 C8PFA4 137356361 IC50 = 37 nM T74312 C8KJ9Z 137479135 IC50 = 536 nM T74312 CVHF30 137479140 IC50 = 1 nM T74312 CK71FM 137628656 Ki = 1.98 nM T74312 C4FLR5 137631588 IC50 = 4.84 nM T74312 C9JK6X 137631909 IC50 = 197 nM T74312 C21ENQ 137633767 IC50 = 117.1 nM T74312 CNX0F9 137634126 IC50 = 37 nM T74312 CHC70D 137634143 IC50 = 1.32 nM T74312 CIKA49 137634942 IC50 = 0.958 nM T74312 CO69DW 137635249 IC50 = 97.4 nM T74312 C4P2IF 137637892 IC50 = 16.9 nM T74312 C4HM1F 137638023 IC50 = 217 nM T74312 CUK8R1 137638801 IC50 = 3.17 nM T74312 CQTF50 137641213 IC50 = 61000 nM T74312 CK3SU9 137641846 IC50 = 0.588 nM T74312 CAE5S9 137641983 IC50 = 0.101 nM T74312 C36KUM 137642749 IC50 = 64000 nM T74312 C30BEJ 137642892 IC50 = 100.3 nM T74312 CEY68J 137644308 IC50 = 33.43 nM T74312 C7KQH8 137644946 IC50 = 60000 nM T74312 COWX42 137645010 IC50 = 128.8 nM T74312 CP91FN 137647445 IC50 = 172 nM T74312 CBS80D 137649459 IC50 = 266.3 nM T74312 CFAY27 137649943 IC50 = 3.78 nM T74312 CNVQ70 137649953 IC50 = 1.56 nM T74312 CEC1O6 137649964 IC50 = 42.38 nM T74312 CM4H0O 137650155 IC50 = 1.03 nM T74312 CS01DK 137650540 IC50 = 359 nM T74312 CK8I5D 137651707 IC50 = 89.2 nM T74312 CLOI26 137651855 IC50 = 1.05 nM T74312 C28QUP 137652864 IC50 = 3275 nM T74312 CW02QJ 137653003 IC50 = 0.13 nM T74312 CLJ67C 137653052 IC50 = 5.36 nM T74312 CD57IP 137655306 IC50 = 2.31 nM T74312 C71HKP 137655481 IC50 = 68000 nM T74312 C17LIA 137655641 IC50 = 2.7 nM T74312 CLQ2G3 137656781 IC50 = 0.34 nM T74312 C0YP9H 137657483 IC50 = 72000 nM T74312 CPV1S9 137658287 IC50 = 2216 nM T74312 CQMB10 137658515 IC50 = 1880 nM T74312 CNR85B 137658530 IC50 = 16.03 nM T74312 C64GHK 137659108 IC50 = 61000 nM T74312 C1XW3M 137659733 IC50 = 76000 nM T74312 C7WHN6 137659742 IC50 = 7.63 nM T74312 CJY76F 137660572 IC50 = 0.32 nM T74312 CM3UF7 137700779 IC50 > 10000 nM T74312 CH6FJ1 138454786 IC50 = 7 nM T74312 CN0X5D 138454787 IC50 = 18.23 nM T74312 CI1D9F 139600335 IC50 = 4 nM T74312 COB9P2 141456067 IC50 = 5200 nM T74312 CYM0K4 141490246 IC50 = 6.13 nM T74312 C34CKN 141523354 IC50 = 5.31 nM T74312 C14IZV 142432627 IC50 = 5 nM T74312 CU6AC8 142432628 IC50 = 19 nM T74312 CI4X1H 142432629 IC50 = 4 nM T74312 CP2ZU6 142432633 IC50 = 3 nM T74312 COYA18 142432636 IC50 = 71 nM T74312 CSH27D 142432637 IC50 = 4 nM T74312 CZ4CT2 142432638 IC50 = 50 nM T74312 C7DW1O 142432639 IC50 = 53 nM T74312 CDU20I 142432642 IC50 = 10 nM T74312 CK64IS 142445421 IC50 = 5 nM T74312 CE84NX 144944001 IC50 = 7513 nM T74312 CO9P7G 145351804 IC50 > 1000 nM T74312 CL4QZ1 145360580 IC50 = 32 nM T74312 CXVF41 145360582 IC50 = 5.24 nM T74312 C3GI7B 145360584 IC50 = 8.2 nM T74312 CGD38P 145360586 IC50 = 255 nM T74312 CIQY42 145360589 IC50 = 347 nM T74312 CX52YL 145360593 IC50 = 3.19 nM T74312 CETO30 145360595 IC50 = 8.74 nM T74312 C8ZXO2 145360601 IC50 = 37.2 nM T74312 C5RA0B 145360613 IC50 = 127 nM T74312 CS6UW5 145360620 IC50 = 27.7 nM T74312 CIK0R8 145360630 IC50 = 22.2 nM T74312 CR31XG 145360635 IC50 = 1.56 nM T74312 C9LI1T 145360638 IC50 = 35.8 nM T74312 CM07EU 145714274 IC50 = 18 nM T74312 C9ISH6 145925685 IC50 = 123 nM T74312 CNK29G 145949498 Ki = 340 nM T74312 C5JP4F 145949566 Ki = 93 nM T74312 CB98HD 145950262 IC50 = 0.66 nM T74312 C6NPE0 145950316 IC50 = 0.47 nM T74312 C2V1MF 145950542 IC50 = 2.53 nM T74312 CFV8U4 145952625 Ki = 63 nM T74312 CUX04Q 145952950 IC50 = 11.31 nM T74312 CV8DJ4 145952962 Ki = 7 nM T74312 COK37P 145953143 Ki > 10000 nM T74312 C3ABQ7 145953222 IC50 = 124 nM T74312 CT0FE4 145953238 IC50 = 3.8 nM T74312 CL6UR2 145953386 Ki = 30 nM T74312 CDBW50 145953650 IC50 = 3.63 nM T74312 CIS8R7 145955252 IC50 = 15.7 nM T74312 CR8O6B 145956516 Ki = 5 nM T74312 CN26GE 145956618 IC50 = 0.66 nM T74312 C7PU6X 145956666 IC50 = 0.73 nM T74312 CSKI41 145956990 IC50 = 3.42 nM T74312 CY54UC 145957309 IC50 = 6.97 nM T74312 CFGK48 145957444 IC50 = 0.95 nM T74312 CEM1D9 145957785 Ki = 100 nM T74312 CJ4FO8 145957807 IC50 = 0.62 nM T74312 CE4VK8 145957843 Ki = 60 nM T74312 C3N1XY 145959793 Ki = 32 nM T74312 C78BGW 145960126 Ki = 64 nM T74312 C1TBX7 145961861 IC50 = 20.51 nM T74312 CJT41L 145962084 IC50 = 770 nM T74312 C8QJS2 145963808 IC50 = 47 nM T74312 CU64FZ 145963919 IC50 = 20 nM T74312 CT9D0I 145964074 IC50 = 2.6 nM T74312 C9BNT0 145964156 IC50 = 35 nM T74312 CIT76X 145964368 IC50 = 16 nM T74312 CIL40C 145964733 IC50 = 5 nM T74312 CKV61O 145964765 IC50 = 29 nM T74312 C02BEJ 145964833 IC50 = 70 nM T74312 C65YWX 145964882 IC50 = 100 nM T74312 CHC3T0 145965031 IC50 > 10000 nM T74312 CP92ZF 145965329 IC50 = 20 nM T74312 C8J3AE 145965430 IC50 = 20 nM T74312 CZV30K 145965543 IC50 = 6 nM T74312 CU2Q9Z 145965567 IC50 = 1141 nM T74312 C8LF7A 145965583 IC50 = 44 nM T74312 CS8DW3 145965618 IC50 = 13 nM T74312 C9HXI4 145966620 IC50 = 530 nM T74312 C4XJ7Z 145966726 IC50 = 23 nM T74312 CQE9M5 145966810 IC50 = 8 nM T74312 C5DY8P 145966963 IC50 = 281 nM T74312 C1EH6C 145967078 IC50 = 250 nM T74312 C1GJ5M 145967083 IC50 = 26 nM T74312 C4OD9Q 145967187 IC50 = 55 nM T74312 CDW83M 145967332 IC50 = 851.8 nM T74312 CDNC31 145967951 IC50 = 5 nM T74312 C5E8ZK 145968310 IC50 = 949 nM T74312 CN6M2H 145968451 IC50 = 1 nM T74312 CHAU61 145968737 IC50 = 67 nM T74312 CWJ12M 145969155 IC50 = 1.4 nM T74312 CGW5S1 145969844 IC50 = 700 nM T74312 CHFQ03 145969846 IC50 = 10 nM T74312 CB8R3A 145970271 IC50 = 300 nM T74312 C5VWH3 145970734 IC50 = 62 nM T74312 C8NK3O 145970839 IC50 = 781 nM T74312 CQO63F 145971860 IC50 = 3.1 nM T74312 C5YKL1 145972178 IC50 = 0.65 nM T74312 CV6IX5 145972308 IC50 = 12 nM T74312 CG59TO 145972635 IC50 > 20000 nM T74312 CS9PM6 145972964 IC50 = 18 nM T74312 C40VIL 145972979 IC50 = 100 nM T74312 CSO3Y9 145973328 IC50 = 6 nM T74312 CX5YI4 145973711 IC50 = 1723 nM T74312 CQBY19 145974023 IC50 > 10000 nM T74312 CTLI02 145974187 IC50 = 4 nM T74312 CGPO78 145974202 IC50 = 4 nM T74312 CXRY95 145974888 IC50 = 950 nM T74312 CZJE72 145974986 IC50 = 628 nM T74312 C74TYP 145975351 IC50 = 2.18 nM T74312 CD7K2U 145975357 IC50 = 591 nM T74312 CMQ64T 145975459 IC50 = 5 nM T74312 CIEM28 145975726 IC50 = 16.5 nM T74312 CY84JV 145976062 IC50 = 4207 nM T74312 C2Q0KP 145976789 IC50 = 10 nM T74312 CC1B8Y 145976973 IC50 = 1195 nM T74312 C4X7CT 145977420 IC50 = 1200 nM T74312 CF49ZG 145977457 IC50 = 25 nM T74312 C2E9WJ 145977590 IC50 = 209 nM T74312 C7Q2KZ 145977606 IC50 = 9848 nM T74312 CMLJ12 145978243 IC50 = 798 nM T74312 CLA57T 145978300 IC50 = 860 nM T74312 C6KDQ5 145979093 IC50 = 3729 nM T74312 C5TP2U 145979643 IC50 = 3800 nM T74312 CV7QY8 145981517 IC50 = 296 nM T74312 CCS92I 145982511 IC50 = 40 nM T74312 CWE21T 145982588 IC50 = 565 nM T74312 CFZ06Y 145982656 IC50 = 1370 nM T74312 CZ3CG9 145982825 IC50 = 311 nM T74312 CRL19G 145983447 IC50 = 5 nM T74312 C48UZH 145983504 IC50 = 128 nM T74312 C8BZC5 145983753 IC50 = 9 nM T74312 CNK7I9 145984104 IC50 = 1010 nM T74312 C4C2OM 145984258 IC50 = 4 nM T74312 C9DHL3 145984282 IC50 = 449 nM T74312 CVT02P 145984555 IC50 = 3 nM T74312 CHW8E5 145984671 IC50 = 191 nM T74312 C4WE0F 145985515 IC50 = 438 nM T74312 C9Q5VI 145985608 IC50 = 51 nM T74312 CV78XO 145985621 IC50 = 1026 nM T74312 C9Y7UN 145985711 IC50 = 39 nM T74312 CA2TW8 145985737 IC50 = 24 nM T74312 CG14RH 145986121 IC50 = 177 nM T74312 C03PYD 145986466 IC50 = 120 nM T74312 CX5MB2 145986730 IC50 = 13790 nM T74312 C1Y5MO 145987062 IC50 = 1.16 nM T74312 CD98JK 145989189 IC50 = 73 nM T74312 CWH69B 145989428 IC50 = 45 nM T74312 CZCS58 145989494 IC50 = 43 nM T74312 CMBH76 145991936 IC50 = 0.9 nM T74312 CNC69T 145992844 IC50 = 2600 nM T74312 C0SO4N 145993259 IC50 = 558 nM T74312 CI7F4G 145994227 IC50 = 51 nM T74312 C7CH9V 146014951 IC50 = 1 nM T74312 CEH17R 153524911 IC50 = 8.422 nM T74312 C1VO9F 153524914 IC50 = 1.518 nM T74312 CZPF13 153524920 IC50 = 4.434 nM T74312 CONR74 154637047 IC50 = 30 nM T74312 C7HKA9 154637067 IC50 = 21 nM T74312 CL9P8H 154637078 IC50 = 30 nM T74312 CYGN68 155510554 IC50 > 10000 nM T74312 C4N1VH 155511342 IC50 = 1.96 nM T74312 CZAB58 155511408 IC50 = 20 nM T74312 CGL79D 155511411 IC50 = 6 nM T74312 CJB1R5 155511461 IC50 = 357 nM T74312 C1WRE2 155511764 IC50 = 15 nM T74312 C1T4ZV 155512315 IC50 = 63.65 nM T74312 C7CA5Q 155512568 IC50 = 4.074 nM T74312 C7X3WN 155513030 IC50 = 4530 nM T74312 C2MD1Q 155513187 IC50 > 10000 nM T74312 C16MVG 155513313 IC50 = 26 nM T74312 C58GHZ 155513629 IC50 = 49 nM T74312 CWG0X8 155513942 IC50 = 1.349 nM T74312 C51BEJ 155514511 IC50 = 9 nM T74312 CTWS76 155514762 IC50 = 123.9 nM T74312 C4PG5Z 155515571 IC50 = 9 nM T74312 CZ7WI9 155515609 IC50 = 70 nM T74312 C9TBG2 155515679 IC50 = 15 nM T74312 CPW74V 155515819 IC50 > 10000 nM T74312 CBZ0T9 155515949 IC50 = 23.44 nM T74312 CVXC96 155516096 Ki = 10.14 nM T74312 CPT39F 155516181 IC50 > 1000 nM T74312 CKMG74 155516483 IC50 > 12500 nM T74312 C0GN6V 155517600 IC50 = 2.042 nM T74312 C4ZSL8 155517778 IC50 = 221.7 nM T74312 CGN7K0 155517959 IC50 = 7.413 nM T74312 C0BC1Z 155518360 IC50 = 200 nM T74312 CE0RN7 155518588 IC50 > 1000 nM T74312 CDM26X 155518680 IC50 = 10.72 nM T74312 C2PBL3 155518730 IC50 > 10000 nM T74312 C5MF1P 155518775 IC50 = 610 nM T74312 C7MBL5 155519087 IC50 = 19.5 nM T74312 C3VTM7 155519139 IC50 = 8.6 nM T74312 C7GAQ9 155519166 IC50 = 61.66 nM T74312 C8EMU7 155519453 IC50 = 1.82 nM T74312 CM51TE 155519497 IC50 = 20 nM T74312 CB4YL6 155519772 IC50 = 6 nM T74312 CP5S9M 155520246 IC50 = 34 nM T74312 CKD52G 155520766 IC50 > 10000 nM T74312 CWQ16B 155521676 IC50 = 32.36 nM T74312 CHP7Q9 155521761 IC50 = 64 nM T74312 C3ST0D 155522792 IC50 = 110 nM T74312 CN5FZ9 155523205 IC50 = 1.318 nM T74312 CXFH76 155523422 IC50 = 4.37 nM T74312 CJKZ10 155523626 IC50 = 2.399 nM T74312 CZ0WO7 155523990 IC50 = 13 nM T74312 CW80OV 155524208 IC50 = 17 nM T74312 C8O2RX 155525008 IC50 = 384 nM T74312 CE15MA 155525223 IC50 = 8.511 nM T74312 CMY37Z 155525462 IC50 = 69 nM T74312 CU7EQ5 155525897 IC50 = 40 nM T74312 CH31QX 155526035 IC50 = 4.365 nM T74312 CIUT60 155526078 IC50 = 47.86 nM T74312 C3INM8 155526137 IC50 = 2.006 nM T74312 CAGM41 155526264 IC50 = 18.2 nM T74312 CQ4XA9 155527433 IC50 > 10000 nM T74312 CDLW94 155527524 IC50 = 13 nM T74312 CICZ14 155527748 IC50 = 6.918 nM T74312 CHL2B9 155528173 IC50 = 4.266 nM T74312 C4LE0G 155528351 IC50 = 151.36 nM T74312 CWG47C 155528371 IC50 = 1.503 nM T74312 C08ITB 155528638 IC50 = 19 nM T74312 CVW07K 155528897 IC50 = 11 nM T74312 C93WSF 155529858 IC50 = 645.65 nM T74312 CDE67Y 155530246 IC50 = 10450 nM T74312 C4Z0FI 155530881 IC50 > 10000 nM T74312 CT9R6V 155530931 IC50 = 13 nM T74312 CU4LS0 155531668 IC50 = 23.99 nM T74312 C8IP7E 155532982 IC50 > 10000 nM T74312 CL8AI2 155533356 IC50 = 113 nM T74312 C3C5HA 155533443 IC50 = 2.773 nM T74312 CEW27M 155533665 IC50 = 3.212 nM T74312 CWGO95 155533831 IC50 = 2 nM T74312 C8HP4G 155534496 IC50 = 39.61 nM T74312 C91KMD 155534710 IC50 = 12.5 nM T74312 CWA1R4 155535707 IC50 = 22 nM T74312 CO9FB7 155535713 IC50 = 9.772 nM T74312 CBE31N 155535715 IC50 = 398.7 nM T74312 CP89CV 155535891 IC50 = 181.97 nM T74312 C35AOY 155536079 IC50 > 10000 nM T74312 CIQ08H 155536349 IC50 = 25.88 nM T74312 C3LC9I 155536820 IC50 = 0.735 nM T74312 CY7Q0U 155537661 IC50 = 17 nM T74312 CK0P8B 155537868 IC50 = 0.327 nM T74312 CQ8UA4 155538384 IC50 > 10000 nM T74312 CTSM92 155538441 IC50 = 4.6 nM T74312 C8T0OS 155539077 IC50 = 1.711 nM T74312 CFEZ25 155539618 IC50 = 17 nM T74312 C0U3RI 155539733 IC50 = 38 nM T74312 CXV14T 155539760 IC50 > 10000 nM T74312 CWBL64 155539811 IC50 = 20 nM T74312 CU35WB 155539873 IC50 = 0.4786 nM T74312 C7HN2I 155540021 IC50 = 46 nM T74312 C0HC7V 155540067 IC50 = 370 nM T74312 CA5I7X 155541030 IC50 = 7393 nM T74312 CYJ16W 155541132 IC50 = 6 nM T74312 CQT69F 155541208 IC50 = 125.89 nM T74312 CP82MK 155541642 IC50 = 3.12 nM T74312 CSET60 155542027 IC50 = 774.7 nM T74312 CY8PB1 155542894 IC50 > 10000 nM T74312 C4MTS0 155543472 IC50 = 8.318 nM T74312 CHD09S 155543566 IC50 = 5 nM T74312 CDA41J 155543682 IC50 = 1.711 nM T74312 C91QLP 155544652 IC50 = 25 nM T74312 C1BVF0 155544897 IC50 = 8.963 nM T74312 C5VHR3 155545392 IC50 = 32 nM T74312 CI41XY 155545477 IC50 = 19.95 nM T74312 C3SH9E 155545928 IC50 = 562.34 nM T74312 C7WC9S 155546415 IC50 = 8.913 nM T74312 CO7ZM2 155546902 IC50 = 12 nM T74312 CQ0HI1 155547040 IC50 = 32 nM T74312 C80JCB 155547115 IC50 > 10000 nM T74312 C7SF2C 155547229 IC50 = 400 nM T74312 C3VX6K 155547248 IC50 = 41 nM T74312 CMRO16 155547287 IC50 = 105 nM T74312 C0H3VE 155548229 IC50 > 1000 nM T74312 C3NDG1 155548730 IC50 = 269.15 nM T74312 CV69KP 155549861 IC50 = 26 nM T74312 CMF0H7 155550304 IC50 = 1.585 nM T74312 CY7LA2 155550601 IC50 = 30 nM T74312 C1UEJ5 155550648 IC50 = 47.86 nM T74312 C4C0ZU 155551393 IC50 > 12500 nM T74312 CJ6P1V 155551489 IC50 = 134.9 nM T74312 CP4IB6 155551544 IC50 = 16 nM T74312 C1P6KR 155551676 IC50 = 158.49 nM T74312 CX2SU8 155552056 IC50 = 9.55 nM T74312 C8BTE5 155552096 IC50 = 312 nM T74312 C9AWP2 155552272 IC50 = 16.98 nM T74312 CQ92ZH 155552526 IC50 = 60 nM T74312 C7AZ9P 155552731 IC50 = 5224 nM T74312 CORH39 155553574 IC50 > 10000 nM T74312 CZFM93 155553628 IC50 = 0.4074 nM T74312 CAZ94Q 155553786 IC50 = 38.9 nM T74312 CH18PL 155553803 IC50 > 10000 nM T74312 CZQM57 155554194 IC50 = 100.45 nM T74312 CNLQ47 155554686 IC50 = 7 nM T74312 CY0AQ3 155555269 IC50 = 4 nM T74312 C1IR7D 155555739 IC50 = 37 nM T74312 C1L8SV 155555805 IC50 = 86 nM T74312 CQ8SE5 155556081 IC50 = 26.92 nM T74312 C3LSW4 155556602 IC50 = 64 nM T74312 CR6B2A 155557324 IC50 = 51 nM T74312 CFZ97J 155557843 IC50 = 349.6 nM T74312 C7HFI8 155558403 IC50 = 9 nM T74312 C1H2RL 155559093 IC50 = 0.3236 nM T74312 CQ7BX0 155559110 IC50 = 1480 nM T74312 CYZU10 155559170 IC50 = 2.138 nM T74312 CM3WR6 155562439 IC50 = 48.31 nM T74312 CGUO53 155562607 IC50 = 10.51 nM T74312 C4RC3O 155562722 IC50 = 2958 nM T74312 CPGH29 155562880 IC50 = 0.7991 nM T74312 CG1Y5D 155563104 IC50 = 7 nM T74312 CUKC08 155563426 IC50 = 9 nM T74312 CV63DM 155563677 IC50 = 12500 nM T74312 C6VU2S 155563700 IC50 = 21 nM T74312 CY51ZP 155563866 IC50 = 13.8 nM T74312 CFY7H2 155564158 IC50 = 1.905 nM T74312 CD2XG9 155564539 IC50 = 7800 nM T74312 C41SIH 155564681 IC50 = 1.66 nM T74312 C0JTS1 155564948 IC50 = 30.12 nM T74312 CDNY29 155565243 IC50 = 842 nM T74312 C7O1SH 155566283 IC50 = 169.82 nM T74312 CJ91SP 155566738 IC50 = 1198 nM T74312 C3QSW0 155567161 IC50 = 31 nM T74312 C85WEG 155567932 IC50 = 103 nM T74312 CI9DP5 155567936 IC50 = 136.1 nM T74312 CJ4GO2 155568394 IC50 = 38 nM T74312 CN79QF 155569564 IC50 = 2.399 nM T74312 C14DIR 16750188 IC50 = 310 nM T74312 C5UI4F 16750189 IC50 = 78 nM T74312 C6JKT9 16750206 IC50 = 880 nM T74312 CYIU14 16750228 IC50 = 29 nM T74312 CX4I6T 16750253 IC50 = 6 nM T74312 CI79TY 16750254 IC50 = 32 nM T74312 CS6UT4 16750288 IC50 = 30 nM T74312 COM3C1 16750290 IC50 = 40 nM T74312 CI67WG 16750292 IC50 = 19 nM T74312 CIGJ63 16750308 IC50 = 31 nM T74312 CL2SY5 16750330 IC50 = 12 nM T74312 CBWO68 49800164 IC50 = 67 nM T74312 C5JYA3 52941420 IC50 = 470 nM T74312 CE5P2I 53363072 IC50 = 49 nM T74312 CTV60O 53363073 IC50 = 70 nM T74312 CD74BW 53363074 IC50 = 38 nM T74312 CU3M8P 53363075 IC50 = 150 nM T74312 C07FTA 53363076 IC50 = 76 nM T74312 C9JX2G 53363150 IC50 = 26 nM T74312 CJ04SF 53363151 IC50 = 140 nM T74312 CO7Z2P 53363152 IC50 = 67 nM T74312 C1T2LY 53363154 IC50 = 22 nM T74312 C9GEA7 53363242 IC50 = 19 nM T74312 CA06ID 53363244 IC50 = 52 nM T74312 CTSP38 53363245 IC50 = 78 nM T74312 CM7BZ3 53363246 IC50 = 15 nM T74312 C0QON7 53363337 IC50 = 8 nM T74312 CU76JB 53363338 IC50 = 92 nM T74312 C2PU3M 53364335 IC50 = 1100 nM T74312 C10FXI 53364337 IC50 = 190 nM T74312 C2U9QE 53364338 IC50 = 170 nM T74312 D00ATA 5908088 IC50 = 350 nM T74312 D00ERW 44444843 Ki > 2481 nM T74312 D00HSJ 10275789 IC50 = 5.15 nM T74312 D00HVA 11624601 Ki > 2500 nM T74312 D00LMG 5281697 IC50 > 10000 nM T74312 D00RIX 5280443 IC50 = 1450 nM T74312 D00YEV 5281605 IC50 > 10000 nM T74312 D01UYI 5281607 IC50 > 10000 nM T74312 D02BXJ 46864270 IC50 = 2 nM T74312 D02NNT 53232451 IC50 = 82 nM T74312 D02OBA 13454380 IC50 = 3600 nM T74312 D03VAA 13393486 IC50 = 1800 nM T74312 D06HVH 54613583 IC50 > 10000 nM T74312 D06QWO 14824655 IC50 > 10 ug.mL-1 T74312 D06UKS 44222958 EC50 = 4800 nM T74312 D07ADX 54764565 IC50 = 4 nM T74312 D07AXL 11098310 IC50 = 600 nM T74312 D07OSK 6419834 IC50 = 4300 nM T74312 D08AIJ 440735 IC50 > 10000 nM T74312 D08GBT 71295845 IC50 = 290 nM T74312 D08HFG 24809764 IC50 > 10000 nM T74312 D09HVH 135566652 IC50 > 10 nM T74312 D09OLH 5330527 IC50 = 3200 nM T74312 D09PTP 57325421 IC50 = 88 nM T74312 D09PUW 13454368 IC50 > 30000 nM T74312 D0A1CM 5281855 IC50 > 40000 nM T74312 D0BW4G 10907042 IC50 = 230 nM T74312 D0C2GE 67161540 IC50 = 0.85 nM T74312 D0CE3R 5312137 IC50 = 8700 nM T74312 D0CM6T 11314340 IC50 = 134 nM T74312 D0D6MH 11617559 IC50 > 13000 nM T74312 D0D7ZL 5330528 IC50 = 890 nM T74312 D0E7VO 59627005 IC50 = 2.1 nM T74312 D0G0KQ 44411967 IC50 = 10000 nM T74312 D0G3SZ 6918469 IC50 = 1.6 ug.mL-1 T74312 D0G3TK 5280863 IC50 = 2320 nM T74312 D0G5YI 10220822 IC50 = 4600 nM T74312 D0H7MF 11500099 IC50 = 2300 nM T74312 D0I3XZ 11601743 IC50 = 40 nM T74312 D0I7QX 44423635 IC50 = 400 nM T74312 D0J3LR 11634725 Ki = 1400 nM T74312 D0L0MZ 13471348 IC50 = 1700 nM T74312 D0L3JR 25212148 IC50 = 8 nM T74312 D0M4QA 56935577 IC50 = 1.3 nM T74312 D0N7AJ 11409972 IC50 = 5.012 nM T74312 D0Q3NG 11715520 Ki > 2500 nM T74312 D0Q4EQ 16742063 IC50 = 4800 nM T74312 D0R2WK 16038120 IC50 = 3 nM T74312 D0R4FM 122850 IC50 > 10000 nM T74312 D0S7IE 11658882 Ki > 2500 nM T74312 D0T3PW 5281672 IC50 = 1690 nM T74312 D0U3NI 53246941 IC50 = 714 nM T74312 D0U3WQ 9817165 IC50 = 1000 nM T74312 D0UN9O 3385203 IC50 = 300 nM T74312 D0US9O 45275255 IC50 = 45 nM T74312 D0V4EX 54760053 IC50 = 2 nM T74312 D0W7TU 947057 IC50 > 50000 nM T74312 D0X6KS 16125109 IC50 = 694 nM T74312 D0X7IC 53340664 IC50 = 149 nM T74312 D0X7JK 1048845 IC50 = 2900 nM T74312 D0XS9E 5330535 IC50 = 570 nM T74312 D0Y0BK 11524144 IC50 < 1 nM T74312 D0Y0ES 3707 IC50 = 33 nM T74312 D0Y1UL 10561847 IC50 = 1800 nM T74312 D0Y4BL 11676971 IC50 = 21 nM T74312 D0Y7HG 5281616 IC50 > 10000 nM T74312 D0Y9GK 16125106 IC50 = 43 nM T74312 D0Z3DW 9179241 IC50 = 3500 nM T74312 D0ZO8Z 4106590 IC50 = 2100 nM T97071 D00ENY 33032 IC50 = 428000 nM T97071 D0Y6UB 10130754 Ki = 0.2 nM T97071 C9RG4D 97663 IC50 > 100000 nM T97071 C7BKY8 164701 IC50 = 438000 nM T97071 C32YSI 185939 IC50 = 2.3 nM T97071 CX2RG7 222467 IC50 = 20000 nM T97071 C0MHV8 252439 IC50 = 43000 nM T97071 CA43YK 455017 IC50 > 100000 nM T97071 CX9FY6 9209550 Ki = 376 nM T97071 C2MG9X 9797132 Ki = 8 nM T97071 CJ94VY 9800545 EC50 = 9.5 nM T97071 CC0VL8 9813818 IC50 = 1400 nM T97071 CHQY81 9818974 IC50 = 200 nM T97071 CK5HF3 9835255 IC50 = 420 nM T97071 CD46GP 9835597 IC50 = 200 nM T97071 C3JE1U 9857135 IC50 = 38 nM T97071 CKV2I5 9858801 IC50 = 140 nM T97071 CPG01H 9860523 IC50 = 40 nM T97071 CUD8C2 9879453 IC50 = 7 nM T97071 C3BT9A 9899009 IC50 = 930 nM T97071 CDXG58 9915884 IC50 = 226 nM T97071 CRLH87 9952075 IC50 = 93 nM T97071 CH4R0F 9966165 Ki = 1 nM T97071 CN58MA 10039522 IC50 = 20000 nM T97071 C9JI5H 10125929 IC50 = 22 nM T97071 CJN79V 10127264 IC50 = 140 nM T97071 CDZ68A 10131651 IC50 = 69 nM T97071 CE5VR7 10192688 IC50 = 1200 nM T97071 CRN1X3 10193222 IC50 = 12000 nM T97071 C0QVK6 10194465 IC50 = 34 nM T97071 CP1T0O 10215518 IC50 = 22 nM T97071 C9UI7D 10219970 Ki = 700 nM T97071 C2ZPA4 10236477 IC50 = 6100 nM T97071 C2U3FM 10309012 IC50 = 94 nM T97071 CVYX42 10309013 IC50 = 22 nM T97071 CH60BG 10333181 IC50 = 15000 nM T97071 CQ2I3N 10448434 IC50 = 12.5 nM T97071 CWH94A 10530644 IC50 > 100000 nM T97071 C45KSB 10582619 IC50 = 2190 nM T97071 CQ67TG 10582644 IC50 = 3080 nM T97071 CRZ23I 10621775 IC50 = 9140 nM T97071 C1WIS7 10627504 IC50 = 3500 nM T97071 C2O3NY 10628412 IC50 = 1340 nM T97071 C6GR1P 10672367 IC50 = 11500 nM T97071 C05RMO 10674948 IC50 = 8980 nM T97071 CIE16L 10694805 IC50 = 4790 nM T97071 C4CJ7P 10694806 IC50 > 30000 nM T97071 C79KAN 10720220 IC50 > 30000 nM T97071 CSQ5T8 10787095 IC50 = 1590 nM T97071 C36NQH 10789375 IC50 > 100000 nM T97071 C38VJN 10813128 IC50 = 24300 nM T97071 C9LY1B 10817849 IC50 = 5840 nM T97071 CGA5L8 10840340 IC50 = 1430 nM T97071 C1JV7A 10933597 IC50 = 185 nM T97071 C0JIG7 11031538 Ki = 30 nM T97071 CLN53E 11069608 IC50 = 3100 nM T97071 C1CEA0 11085481 Ki = 0.1 nM T97071 C1I4NB 11134118 IC50 > 10000 nM T97071 C61AQD 11321189 IC50 = 1300 nM T97071 CYG85O 11357165 IC50 = 0.86 nM T97071 C28AXU 11364061 Ki = 392 nM T97071 C4TEO7 11416756 Ki = 1109 nM T97071 C6RUL8 11484828 Ki = 1285 nM T97071 CTBL43 11536480 IC50 > 20000 nM T97071 CZ70LS 11569764 IC50 > 20000 nM T97071 CSHC02 11587262 IC50 = 730 nM T97071 CIA80J 11597620 IC50 = 2400 nM T97071 CST94M 11601614 IC50 = 2700 nM T97071 C56XYT 11722553 IC50 = 0.5 nM T97071 C1ZRG0 21915695 IC50 = 2000 nM T97071 CW0M2Q 24951652 Ki = 0.003 nM T97071 CB0YO2 24951653 IC50 = 43 nM T97071 C0Q5NM 24951654 IC50 = 1200 nM T97071 C1PG3H 24951655 IC50 = 22 nM T97071 C4X1VR 24951656 IC50 = 443 nM T97071 CY91LZ 24951657 IC50 = 37 nM T97071 CILH68 24952014 Ki = 44.3 nM T97071 CL2QW9 24953090 IC50 = 245 nM T97071 COD9H3 24953091 IC50 = 277 nM T97071 CH1DJ4 24953092 IC50 = 2 nM T97071 C4VM2H 24953441 IC50 = 2960 nM T97071 CHM36W 24953442 IC50 = 12 nM T97071 CV3L9W 24953443 IC50 = 2 nM T97071 CWS91Q 24953444 IC50 = 4 nM T97071 C76JDG 24953445 IC50 = 154 nM T97071 CTL98E 24953446 IC50 = 18 nM T97071 C35FES 24957010 IC50 = 10 nM T97071 C0RZF3 24957011 IC50 = 10 nM T97071 C6XFR4 25178768 Ki = 0.194 nM T97071 CU9RQ2 25178941 Ki = 0.351 nM T97071 CNS3O2 25194656 IC50 = 3 nM T97071 CKPW37 25194768 IC50 > 3000 nM T97071 C4QDR7 44291751 IC50 = 1340 nM T97071 C9T8FO 44306373 IC50 > 100000 nM T97071 C4Z2UT 44306478 IC50 > 100000 nM T97071 CME60R 44437842 IC50 = 35 nM T97071 C0UTB1 44437850 IC50 = 55 nM T97071 C06TRE 44437852 IC50 = 1800 nM T97071 C5VZU6 44437853 IC50 = 280 nM T97071 CW7VS9 44437854 IC50 = 700 nM T97071 CE13VL 44437856 IC50 = 790 nM T97071 C54JKC 44437858 IC50 = 4100 nM T97071 CD6X7U 44437865 IC50 = 180 nM T97071 CN9AC2 44437871 IC50 = 15 nM T97071 C3DY5U 44455907 IC50 = 569 nM T97071 CSZ25Y 44455939 IC50 = 572 nM T97071 C37EWO 44455941 IC50 = 435 nM T97071 C2KUC3 44455974 IC50 = 140 nM T97071 C1ZL5D 44456014 IC50 = 125 nM T97071 C7B9VK 44456016 IC50 = 438 nM T97071 CP57NB 44456602 IC50 = 4 nM T97071 CG4F0C 44468183 Ki = 11 nM T97071 CPY07J 44604932 IC50 = 9 nM T97071 C2JF1E 44604934 IC50 = 23 nM T97071 C0LHU3 46227558 Ki = 153 nM T97071 C5NS8F 46227559 Ki = 13000 nM T97071 CA7YC4 46227560 Ki > 1000000 nM T97071 CUR58O 46227562 Ki = 3000 nM T97071 CU7C2F 46227568 Ki > 1000000 nM T97071 C7VLX8 46227569 Ki = 81 nM T97071 C1RN8X 46227570 Ki > 1000000 nM T97071 C2ABL6 46227575 Ki = 775 nM T97071 C3K2RP 46227576 Ki = 13000 nM T97071 C2PS0E 46227580 Ki = 3500 nM T97071 COR76U 46227587 Ki = 475 nM T97071 CMZL17 46227590 Ki > 1000000 nM T97071 CF3O2J 46227591 Ki = 7500 nM T97071 CS48DI 46227595 Ki = 250 nM T97071 CBE7J1 46227601 Ki = 275 nM T97071 CT29AQ 46227602 Ki > 1000000 nM T97071 C06FKR 46227609 Ki = 400 nM T97071 CS6L4K 46227610 Ki = 1320 nM T97071 CA26FD 46227611 Ki = 575 nM T97071 C1U0RX 46227612 Ki = 3430 nM T97071 C9F1MO 46227613 Ki = 318 nM T97071 C1ZL2O 46227617 Ki = 3000 nM T97071 CV1I6N 46227618 Ki > 1000000 nM T97071 CL84FP 46227623 Ki = 700 nM T97071 CG2WA8 46227629 Ki > 1000000 nM T97071 C91UCR 46228323 Ki = 23 nM T97071 CQ3KC9 46228324 Ki = 24.1 nM T97071 C79UVH 46228331 Ki = 5.3 nM T97071 C5A8HD 46228334 Ki = 85.1 nM T97071 CP18GF 46228337 Ki = 52.3 nM T97071 CK6BO4 46228340 Ki = 285 nM T97071 CS60AE 46228341 Ki = 5.3 nM T97071 CR9AN1 46228346 Ki = 254 nM T97071 CDLM54 46228347 Ki = 132 nM T97071 CWA1Z5 46228350 Ki = 16.2 nM T97071 CD9J3O 46228351 Ki = 794 nM T97071 C9LNJ1 46228352 Ki = 795 nM T97071 CB6HE9 46228353 Ki = 16.1 nM T97071 C1K2DN 46228356 Ki = 320 nM T97071 C8BIL9 46228364 Ki = 105 nM T97071 C3MNA9 46228365 Ki = 97.2 nM T97071 C0WB2Z 52940848 IC50 = 144 nM T97071 CA5QD0 52941224 IC50 = 24000 nM T97071 CDL1U6 52942433 IC50 = 20000 nM T97071 C92SZW 52943734 IC50 = 54 nM T97071 CWK38S 52944436 IC50 = 6100 nM T97071 CYU68W 52948774 IC50 = 0.55 nM T97071 CT52BD 52949740 IC50 = 1700 nM T97071 C6O5TZ 53250307 Ki = 1.4 nM T97071 CYF19B 53250308 Ki = 3.1 nM T97071 C6MVX1 56643458 Ki = 29 nM T97071 CVA52S 56648026 Ki = 325 nM T97071 CY0LE3 56648027 Ki = 121 nM T97071 C17OTD 56648028 Ki = 56 nM T97071 C7ZMD5 56648117 Ki = 20 nM T97071 C2E3QO 56648118 Ki = 72 nM T97071 C05TFC 57392577 IC50 = 0.35 nM T97071 CS8V1T 57394302 IC50 = 14 nM T97071 C6M5TO 57396056 IC50 = 0.41 nM T97071 CNZH82 57401271 IC50 = 1.93 nM T97071 CE4C2I 60143283 Ki = 0.018 nM T97071 C6FV5R 60148557 IC50 = 2 nM T97071 CWV7X2 60167144 IC50 = 5700 nM T97071 CCER72 60167145 IC50 = 340 nM T97071 C2IS0P 60167146 IC50 = 52 nM T97071 CS6B7I 60167288 IC50 = 41 nM T97071 CI9V4L 60167289 IC50 = 16 nM T97071 CBF10D 60167291 IC50 = 230 nM T97071 CK74OW 71451806 Ki = 36.4 nM T97071 CK17XN 71451807 Ki = 2.6 nM T97071 CYPQ06 71455354 Ki = 22 nM T97071 CETK98 71532123 IC50 = 1.56 nM T97071 CBF45S 72713178 Ki = 4.97 nM T97071 CCAX87 72713180 Ki = 2.79 nM T97071 CJHP02 72713181 Ki = 62.1 nM T97071 CF85HT 72713391 Ki = 94.8 nM T97071 C01TXM 72713394 Ki = 8.06 nM T97071 C7OU1Q 72713617 Ki = 7.91 nM T97071 C59KEM 72713848 Ki = 6.26 nM T97071 C0E4XS 72713849 Ki = 2.95 nM T97071 C2R8KP 72713850 Ki = 2.14 nM T97071 CO62TF 73386645 IC50 = 400 nM T97071 CFI74Y 74627713 Ki = 0.0449 nM T97071 C8NX3I 74627717 Ki = 0.268 nM T97071 C7IE3R 74627718 Ki = 0.377 nM T97071 C67ABM 74627719 Ki = 0.221 nM T97071 C93HNS 86297087 IC50 = 19000 nM T97071 CM1G4Y 86306042 IC50 = 1300 nM T97071 CQH50K 89819943 Ki = 0.17 nM T97071 C2PR8X 89986823 IC50 = 3 nM T97071 CQD2I7 89986839 IC50 = 123 nM T97071 CD5YJ9 90447523 IC50 = 27000 nM T97071 C03HER 92460914 IC50 = 15.9 nM T97071 C3A2KL 118706009 Ki = 6.39 nM T97071 C1QY5B 118706010 Ki = 10.5 nM T97071 C4W9EQ 118706011 Ki = 1.58 nM T97071 CKD32U 118706012 Ki = 28.1 nM T97071 CY9GE4 118706013 Ki = 7.6 nM T97071 C7GBS1 118706014 Ki = 0.312 nM T97071 CSB65R 118706015 Ki = 3.42 nM T97071 C16HUL 118706016 Ki = 0.601 nM T97071 CELI50 118706017 Ki = 10.97 nM T97071 C2F4KE 118706018 Ki = 1.012 nM T97071 CTAH37 118706019 Ki = 0.722 nM T97071 C5Y1FB 118706020 Ki = 0.6 nM T97071 CN1RD9 118706021 Ki = 1.57 nM T97071 C9IK6Q 118706022 Ki = 3.88 nM T97071 C36DPO 118737810 IC50 = 60000 nM T97071 CPO7F2 118737811 IC50 = 357000 nM T97071 CB28DM 118737812 IC50 = 79000 nM T97071 C69RFT 118737813 IC50 = 112000 nM T97071 CK36FN 118737814 IC50 = 2600 nM T97071 CL2G4Q 118737815 IC50 = 3000 nM T97071 C9Y2IL 118737816 IC50 = 1300 nM T97071 CBM15Z 118737817 IC50 = 11000 nM T97071 CC79YB 118987236 IC50 = 97 nM T97071 C0DU8Y 118987238 IC50 = 44 nM T97071 CO1X5J 122178329 Ki = 0.071 nM T97071 CQA5H4 122178330 Ki = 1.6 nM T97071 C6KUH2 122178331 Ki = 0.049 nM T97071 CEU7B1 122178332 Ki = 0.11 nM T97071 CRY6O0 122178333 Ki = 0.0086 nM T97071 CDK0O7 127031340 IC50 = 30 nM T97071 CNKT62 127031341 IC50 = 24 nM T97071 C9DA8S 127031342 IC50 = 15 nM T97071 CG0VX5 127031620 IC50 = 14 nM T97071 C7J2UN 127032189 IC50 = 19 nM T97071 C2IL3O 127032190 IC50 = 98 nM T97071 C5R8BC 132160022 IC50 = 16.9 nM T97071 C3EAX0 132160242 IC50 > 1000 nM T97071 CWO5G1 134130685 IC50 = 28 nM T97071 CBRW84 134524274 IC50 > 5000 nM T97071 CJ06BW 134533331 IC50 = 540 nM T97071 CC37ZL 134533335 IC50 > 5000 nM T97071 CU51BV 134533356 IC50 > 5000 nM T97071 CMQA75 134533371 IC50 > 5000 nM T97071 CL28JY 134533387 IC50 > 5000 nM T97071 CGQ41D 134693711 IC50 = 2.32 nM T97071 CE40DB 134823841 IC50 = 8.9 nM T97071 C2RX7B 135121378 IC50 = 0.35 nM T97071 CSR16B 135121379 IC50 = 0.075 nM T97071 CJBX90 135121380 IC50 = 0.99 nM T97071 C4M2XI 135121381 IC50 = 0.13 nM T97071 C9AR8E 135121924 IC50 = 0.65 nM T97071 CYJQ73 145949136 IC50 = 25 nM T97071 CIK62H 145964139 Ki = 0.14 nM T97071 C5SPF7 145976481 Ki = 0.58 nM T97071 C27ICA 145976922 Ki = 0.38 nM T97071 C7F5VX 145978984 IC50 = 5.24 nM T97071 C4PE1V 145979935 IC50 = 1.19 nM T97071 C0CP2G 145981270 IC50 = 4.46 nM T97071 C9N5IM 145982923 IC50 = 0.28 nM T97071 C9FCU1 145986913 IC50 = 1.11 nM T97071 CKY98A 145989288 IC50 = 1.31 nM T97071 C5QT1C 145989357 IC50 = 0.46 nM T97071 C6R1OY 145990708 IC50 = 5.44 nM T97071 C6PN9S 145991345 IC50 = 2.91 nM T97071 C2RZ5O 145991423 IC50 = 0.64 nM T97071 C7JY5R 145991877 IC50 = 0.2 nM T97071 CZ6R8C 145993125 IC50 = 0.15 nM T97071 C9E2CQ 145993836 IC50 = 2.11 nM T97071 C7LY6Q 145994234 IC50 = 0.94 nM T97071 C09WTD 146035548 IC50 = 3.97 nM T97071 CFOA50 146035557 IC50 = 107 nM T97071 CBVG30 149751695 IC50 > 1000 nM T97071 CS6JN2 149751696 IC50 = 399 nM T97071 CR3WN8 150793150 IC50 = 155 nM T97071 CBZ10S 150793151 IC50 = 16.7 nM T97071 CO91TE 152021787 IC50 = 11 nM T97071 CU17ZK 152577625 IC50 = 11.9 nM T97071 CDJI50 152577626 IC50 > 1000 nM T97071 CZ90MS 152682917 IC50 = 284 nM T97071 CW23PU 152682918 IC50 > 1000 nM T97071 CZ79UN 153564422 IC50 > 1000 nM T97071 CR2DN1 153564423 IC50 = 195 nM T97071 CW7ZE3 153564425 IC50 > 1000 nM T97071 C6NH4B 153564426 IC50 > 1000 nM T97071 CCZ18P 155517395 IC50 = 140 nM T97071 CVB6M3 155520777 IC50 = 170 nM T97071 CIR93U 155523285 IC50 > 1000 nM T97071 C5MQD2 155529343 IC50 = 630 nM T97071 C1H2XP 155529636 IC50 = 110 nM T97071 CDE4B6 155538994 IC50 = 8530 nM T97071 C0S2RH 155567546 IC50 = 531 nM T97071 D02CYQ 20778210 IC50 = 4000 nM T97071 D03JFL 44410794 IC50 = 190 nM T97071 D03RMT 11666341 IC50 = 390 nM T97071 D04SMQ 440053 IC50 = 67000 nM T97071 D04SZR 9878511 IC50 = 63 nM T97071 D04VFS 11615808 IC50 = 1100 nM T97071 D05SNS 20778197 IC50 = 1200 nM T97071 D05VWZ 11499788 IC50 = 15000 nM T97071 D06DUE 40539 IC50 = 9500 nM T97071 D07CVG 194327 Ki = 11 nM T97071 D07PZQ 68841 IC50 = 523000 nM T97071 D08CYU 10171263 IC50 = 2600 nM T97071 D08TDE 10130679 IC50 = 1100 nM T97071 D0A1FL 11020196 IC50 = 1400 nM T97071 D0B9YO 9920926 IC50 = 1400 nM T97071 D0C2FS 9794137 IC50 = 580 nM T97071 D0C5JP 11492994 IC50 = 120 nM T97071 D0D8NM 11601420 IC50 = 2200 nM T97071 D0E0HK 129558 IC50 = 6000 nM T97071 D0E3OH 11715765 IC50 = 1800 nM T97071 D0F8TZ 9878510 IC50 = 15 nM T97071 D0FU7Y 10219893 EC50 = 220 nM T97071 D0G9LM 449178 IC50 > 100000 nM T97071 D0JX2S 11694647 IC50 = 640 nM T97071 D0ND1C 9900104 IC50 = 14 nM T97071 D0Q2OH 11790725 IC50 = 6500 nM T97071 D0Q3KD 10955499 IC50 = 2600 nM T97071 D0QA5U 9921539 IC50 = 1700 nM T97071 D0T8ZL 11557761 IC50 = 440 nM T97071 D0X1DO 11666386 IC50 = 32 nM T97071 D0Y7AN 10198171 EC50 = 13 nM T97071 D0Z0UQ 10909614 IC50 = 1400 nM T97071 D0Z5VI 10879227 IC50 = 1200 nM T97071 D0ZJ9S 20778204 IC50 = 940 nM T26220 D09YDM 24360 IC50 = 2.21 nM T26220 D08AWI 11430856 Ki > 2000 nM T26220 CW7I8U 13690207 IC50 = 1.1 nM T26220 C7K5AW 16721015 IC50 > 10000 nM T26220 CPK4L5 44278770 IC50 = 0.46 nM T26220 C3XOA2 44403691 IC50 = 14000 nM T26220 CRCO43 44403692 IC50 = 5100 nM T26220 CP8JT3 44403693 IC50 = 8400 nM T26220 C91HUQ 44403694 IC50 = 6600 nM T26220 CW0O6U 44403695 IC50 = 10000 nM T26220 CORN26 44403697 IC50 = 34000 nM T26220 CU3PS6 44403698 IC50 = 35000 nM T26220 CRSP62 44403699 IC50 = 47000 nM T26220 CJ4UE0 44420802 IC50 = 0.2 nM T26220 CO0P5S 44420803 IC50 = 0.64 nM T26220 CMOQ24 44420804 IC50 = 0.5 nM T26220 C0Y3PV 44420805 IC50 = 1.6 nM T26220 CK17OQ 44420806 IC50 = 0.35 nM T26220 CXJF19 44420807 IC50 = 1.6 nM T26220 C4MT8I 56681776 IC50 = 15000 nM T26220 CY1ZQ6 71715991 IC50 = 15000 nM T26220 C4BUD8 71717816 IC50 = 11000 nM T26220 C0CQZ9 73345571 IC50 = 2.79 nM T26220 C2HQ7A 73348598 IC50 > 1000 nM T26220 CU18EB 73348599 IC50 = 54.2 nM T26220 CYBE03 73348600 IC50 = 571 nM T26220 C3BNZ8 73351683 IC50 > 1000 nM T26220 D0T5RO 16129706 IC50 = 0.83 nM T80896 D00ZFP 5870 EC50 = 2.1 nM T80896 D01XBA 5035 Ki = 2.74 nM T80896 D06LOQ 179337 IC50 = 240 nM T80896 D06NXY 5991 IC50 = 8.1 nM T80896 D06XMU 6013 IC50 > 10000 nM T80896 D07BSQ 5994 IC50 1000000 nM T80896 D07KSG 2733526 Ki = 0.51 nM T80896 D08QMX 5757 EC50 = 0.01 nM T80896 D09NMD 216416 IC50 = 1.8 nM T80896 D0D1SG 5755 IC50 > 10000 nM T80896 D0EP0C 5833 EC50 = 3300 nM T80896 D0JO7Y 104741 Ki = 1.39 nM T80896 D0JY8T 154257 IC50 = 3.8 nM T80896 D0Q4SD 443872 EC50 > 20000 nM T80896 D0Y2NE 448537 EC50 = 0.02 nM T80896 D0Y7IU 5281004 IC50 > 10000 nM T80896 D0Y7JU 9854489 IC50 > 5000 nM T80896 D0Z1FX 5756 EC50 = 0.1259 nM T80896 D0Z4EI 55245 Ki > 750 nM T80896 D00JFE 56941241 IC50 = 8.8 nM T80896 D07LZH 656954 IC50 = 5 nM T80896 D0L4FS 5280961 EC50 = 1.7 nM T80896 D0LI1C 44469321 IC50 > 30000 nM T80896 D0R2SK 10286159 Ki = 0.17 nM T80896 D0SZ1G 121248172 IC50 > 100000 nM T80896 D0X9YP 67041274 IC50 > 10000 nM T80896 D05BCA 68570 EC50 = 4.5 nM T80896 D08DZZ 10634 EC50 = 5.6 nM T80896 D08HIH 6102691 IC50 = 2.7 nM T80896 D09UFV 24825740 IC50 > 10000 nM T80896 D0H5CV 130936 IC50 = 242 nM T80896 D0R8TB 6433099 IC50 = 40 nM T80896 D0U7OU 3220 Ki = 1500 nM T80896 C3EUZ1 6776 Ki = 690 nM T80896 C2SL4X 7074 IC50 = 3100 nM T80896 C6QYD8 8434 EC50 = 1860 nM T80896 CHA7C3 12111 EC50 = 1900 nM T80896 CGWM38 54900 IC50 = 43 nM T80896 CSI62C 62082 EC50 = 1.2 nM T80896 CQ0IC4 63062 Ki = 0.014 nM T80896 C38RAY 65434 EC50 = 72 nM T80896 CF5JU9 75386 IC50 = 790 nM T80896 CYCI69 80152 EC50 = 9.3 nM T80896 CNT0H1 96201 IC50 = 270 nM T80896 CS8Q6W 99649 Ki = 18000 nM T80896 C5E2IG 223998 Ki = 24 nM T80896 C78YGO 232446 IC50 = 560 nM T80896 C8MJB2 247310 IC50 = 770 nM T80896 CDHI70 251929 EC50 = 210 nM T80896 C9XC2A 252281 IC50 > 10000 nM T80896 CDP78A 261349 IC50 = 9.4 nM T80896 C7HME8 439246 IC50 = 13473 nM T80896 C5SEF1 442342 IC50 1000000 nM T80896 C40YBS 444036 IC50 > 10000 nM T80896 CJZO27 445920 Ki = 2.3 nM T80896 CK01NI 448577 IC50 = 45 nM T80896 CGT37O 449205 IC50 = 37 nM T80896 C9AXQ3 449207 IC50 = 22 nM T80896 CBD7O2 449208 IC50 = 45 nM T80896 CL26SB 449209 IC50 = 45 nM T80896 CMT3P0 480764 EC50 = 5 nM T80896 C0CF9H 586500 IC50 = 43000 nM T80896 CZ0AH3 638278 IC50 = 269 nM T80896 C9UW8R 640096 EC50 = 500 nM T80896 C2I3PM 646429 EC50 = 1460 nM T80896 CB20EC 656952 IC50 = 2.2 nM T80896 C67LKM 656953 IC50 = 14 nM T80896 CX8H6W 687290 EC50 = 4070 nM T80896 C3R1PZ 721251 IC50 1000000 nM T80896 C1OG7J 833976 EC50 = 34900 nM T80896 CV95AN 837745 EC50 = 13400 nM T80896 C31BFY 837746 EC50 = 8590 nM T80896 C69DLW 837838 IC50 > 100000 nM T80896 C4T6YS 837853 IC50 > 100000 nM T80896 C06JQG 837872 EC50 = 4950 nM T80896 CQOD41 837886 EC50 = 485 nM T80896 C1ZE2H 845978 IC50 = 180 nM T80896 C6XGH8 849252 IC50 = 1520 nM T80896 C9S4EA 849257 IC50 = 2820 nM T80896 CE9VY2 849282 EC50 = 2690 nM T80896 C4IQG9 849291 EC50 = 185 nM T80896 CN6RA2 849298 EC50 = 823 nM T80896 CPQ72T 849308 IC50 = 3910 nM T80896 C45RBT 851153 EC50 = 7060 nM T80896 CO85AF 902564 EC50 = 28900 nM T80896 C5MZH8 906479 IC50 = 4480 nM T80896 C2LRG9 927532 EC50 = 195 nM T80896 C5A7CD 928630 IC50 1000000 nM T80896 C90CUZ 1111980 EC50 > 10000 nM T80896 C5GJF1 1234611 IC50 = 8940 nM T80896 CM6NY1 1234663 IC50 = 4350 nM T80896 CMBE67 1234708 IC50 = 1310 nM T80896 C7TE0L 1717570 EC50 = 5770 nM T80896 CF4S1M 1731992 EC50 = 94 nM T80896 C8WS4M 2040507 IC50 1000000 nM T80896 CLF0C9 2288503 IC50 = 93 nM T80896 CS6TF7 2733525 IC50 = 5 nM T80896 C6LXG3 2747677 IC50 = 300 nM T80896 CFH19O 2887782 IC50 = 6200 nM T80896 CJ6Z8I 2999413 EC50 = 24 nM T80896 CBZ6U1 3024714 IC50 = 421 nM T80896 C7RNA9 3325226 IC50 = 289 nM T80896 C9S2LO 4055843 EC50 = 894 nM T80896 C6J0ZF 4369568 IC50 = 12 nM T80896 CFY94M 4369569 IC50 = 18 nM T80896 C0N9SD 4598916 EC50 = 19000 nM T80896 CMB6I1 5281576 EC50 = 110 nM T80896 CH6RY7 5282240 EC50 = 3.6 nM T80896 CB6OK2 5287464 IC50 = 3.5 nM T80896 C7IBX9 5287551 IC50 = 1 nM T80896 CJB7T6 5288494 IC50 = 56 nM T80896 CW91XD 5322257 EC50 = 46.3 nM T80896 CS31LU 5322291 EC50 = 71 nM T80896 CP69KZ 5324349 IC50 = 1.7 nM T80896 C2JOL1 5327043 Ki = 1.32 nM T80896 CN7CS6 5372367 IC50 = 286.5 nM T80896 CF5VB6 5395460 IC50 1000000 nM T80896 C9GS2K 5397219 EC50 = 33.8 nM T80896 CQ83GI 5397398 IC50 1000000 nM T80896 C4Z1IB 5400235 EC50 = 67.2 nM T80896 CNG5W4 5407968 IC50 = 308 nM T80896 CO36YU 5455071 EC50 = 5360 nM T80896 C52EHD 5822393 EC50 = 3910 nM T80896 CY9MR6 5885714 IC50 = 49.7 nM T80896 CT0F6H 5948122 IC50 = 250 nM T80896 C6LCX3 6260040 EC50 = 49.8 nM T80896 CL41HW 6303362 EC50 = 140 nM T80896 C6RDY2 6444422 EC50 = 2.21 nM T80896 C3E0BP 6604873 EC50 = 0.8 nM T80896 CF61LI 7314046 EC50 = 229 nM T80896 CM5Y0Z 7314049 IC50 = 2670 nM T80896 CXHO01 7314090 EC50 = 1980 nM T80896 CFM7Q8 7314234 EC50 = 1010 nM T80896 C3M7RE 9804246 IC50 = 2049 nM T80896 CU3QR8 9808162 Ki = 8 nM T80896 CE23GX 9814262 IC50 = 31.8 nM T80896 C34IZS 9814547 IC50 = 5.3 nM T80896 CZA2O0 9814673 IC50 = 11 nM T80896 CCUR98 9815144 IC50 = 23 nM T80896 CTB3F6 9815173 IC50 = 21 nM T80896 CNJK98 9816989 Ki = 47 nM T80896 CX1F7P 9819159 IC50 = 11.4 nM T80896 CTXR52 9820272 EC50 > 100000 nM T80896 CN9M3P 9824019 Ki = 3.2 nM T80896 C94INP 9829162 IC50 = 1500 nM T80896 C7V2ZD 9835427 EC50 = 5 nM T80896 CCX60E 9835779 IC50 = 12 nM T80896 CS97CD 9846731 IC50 = 1.9 nM T80896 C2LV3C 9848252 IC50 = 38 nM T80896 CMI0N6 9848501 Ki = 0.48 nM T80896 CQGZ49 9856356 EC50 = 76 nM T80896 CVW25C 9856632 EC50 = 20 nM T80896 C8ER6V 9869745 Ki = 200 nM T80896 C9MA0B 9878811 EC50 = 1.7 nM T80896 CIA6K1 9878841 EC50 = 7.3 nM T80896 CJ8VH6 9879228 EC50 = 20 nM T80896 CPF25S 9879409 IC50 = 42.5 nM T80896 CA1CJ6 9879798 EC50 = 30 nM T80896 C01ZFV 9882789 IC50 > 10000 nM T80896 CIT93X 9884138 IC50 = 1.8 nM T80896 CL8E7Z 9890509 IC50 = 136 nM T80896 CL7UB1 9900112 IC50 = 20 nM T80896 C3EQA8 9900383 EC50 = 17 nM T80896 C30BCU 9900479 EC50 = 2 nM T80896 CM9S2I 9900695 IC50 = 13.4 nM T80896 C3C6GN 9902151 EC50 = 5 nM T80896 C2BUL1 9902785 EC50 = 18 nM T80896 CLC48G 9909681 IC50 = 1.21 nM T80896 CCZ9P8 9911175 Ki > 10000 nM T80896 CD3A6G 9912022 Ki = 4.4 nM T80896 C6YGM0 9912245 IC50 = 1404 nM T80896 C58PVC 9921352 IC50 = 11 nM T80896 CJL2P9 9921784 IC50 = 12.6 nM T80896 CBX75P 9922298 IC50 = 1.5 nM T80896 CGN5C8 9922681 IC50 = 43 nM T80896 CX9AV7 9923647 EC50 = 46 nM T80896 CJD4H0 9923941 IC50 = 1.6 nM T80896 CFT7M0 9924049 IC50 = 5.9 nM T80896 C9I3SQ 9924986 IC50 = 4.9 nM T80896 CE6HU3 9925763 Ki = 0.47 nM T80896 CP8ZG3 9927355 Ki = 0.28 nM T80896 CVW4Y8 9935633 IC50 = 9.6 nM T80896 CB0H3V 9942858 IC50 = 28 nM T80896 CB65XA 9943599 IC50 = 283 nM T80896 CW4RV2 9945087 EC50 = 96 nM T80896 CO4IM2 9946131 IC50 = 5.4 nM T80896 C81CGQ 9946229 EC50 = 6.5 nM T80896 CZP05L 9948127 Ki = 0.31 nM T80896 CQ04ES 9948426 IC50 = 128 nM T80896 CY6M2H 9953602 IC50 = 22.2 nM T80896 C9OPU4 9957008 IC50 = 6 nM T80896 CO5V0P 9964601 IC50 = 63 nM T80896 C0AJ3H 9964943 EC50 = 475 nM T80896 CJT98P 9965271 EC50 = 20 nM T80896 C0LGC8 9965955 EC50 = 7.7 nM T80896 C1ZBV6 9967036 EC50 = 40 nM T80896 C29KIM 9968828 IC50 = 1.8 nM T80896 C4XGS5 9970588 Ki = 11 nM T80896 C05NAQ 9973567 IC50 = 22 nM T80896 COJ0E4 9993475 IC50 = 21 nM T80896 CB6AC7 10002045 IC50 = 31 nM T80896 CDU28H 10005346 IC50 = 134 nM T80896 CW4B6F 10015172 IC50 = 80 nM T80896 CJN7T4 10016716 IC50 = 16 nM T80896 C3XCR4 10016731 IC50 = 2.3 nM T80896 C7NLS3 10016946 EC50 = 190 nM T80896 C8UT2P 10019713 IC50 = 433 nM T80896 CG8B1H 10026593 IC50 = 82 nM T80896 C30UFB 10028024 IC50 = 87 nM T80896 CE0X1Y 10038212 IC50 = 54 nM T80896 CSA35D 10051476 IC50 = 5.3 nM T80896 C2WYO1 10060623 EC50 = 1100 nM T80896 C3QBA5 10060912 IC50 = 279 nM T80896 C9Z0AT 10060945 EC50 = 7.2 nM T80896 CIY1Z7 10064013 IC50 = 18 nM T80896 C37ZQE 10072011 Ki = 190 nM T80896 C8P1BZ 10084254 IC50 = 116 nM T80896 CDM8V3 10084479 IC50 = 5.7 nM T80896 CT1ZO9 10085265 EC50 = 1583 nM T80896 CYH2U5 10086047 IC50 = 49 nM T80896 CMDP60 10107798 IC50 = 53 nM T80896 CM4B3Q 10108320 IC50 = 14.3 nM T80896 C96JZH 10113416 IC50 = 42.2 nM T80896 C4XU7H 10115709 IC50 = 50 nM T80896 C9EDV6 10115710 IC50 = 48 nM T80896 CCA85G 10125282 IC50 = 11 nM T80896 CWLS93 10125319 IC50 = 81 nM T80896 CTF5J0 10125414 Ki = 0.66 nM T80896 CH4N0B 10125582 IC50 = 32 nM T80896 CYIT90 10125667 IC50 = 10 nM T80896 CRP1U3 10128287 IC50 = 21 nM T80896 C08BYF 10140504 IC50 = 73 nM T80896 CQK5X9 10144672 Ki = 35 nM T80896 CC24WL 10149300 IC50 = 847 nM T80896 CO1AE6 10149393 IC50 = 32 nM T80896 C8G4PV 10149522 IC50 = 8 nM T80896 CY15UJ 10149610 IC50 = 8.5 nM T80896 C2EOX1 10151898 IC50 = 1.3 nM T80896 CIEH85 10154586 EC50 = 1.5 nM T80896 C1BAI4 10171529 Ki = 22.1 nM T80896 CT5W0A 10171640 IC50 = 3 nM T80896 CD36GZ 10171641 IC50 = 1.3 nM T80896 C36ACW 10171666 IC50 = 4 nM T80896 C5I7DH 10171723 Ki = 0.63 nM T80896 C9P4CF 10171732 IC50 = 58 nM T80896 C5DSH0 10171830 IC50 = 2.5 nM T80896 C3QR7A 10171898 IC50 = 9 nM T80896 CK0ZU9 10172081 IC50 = 267 nM T80896 C1VDO4 10174471 IC50 = 66.6 nM T80896 CJO0M8 10174620 IC50 = 19 nM T80896 CB5J9S 10176498 EC50 = 7520 nM T80896 C2YRA6 10177915 EC50 = 2 nM T80896 C2BS8L 10181886 Ki = 4 nM T80896 CWCM45 10182934 Ki = 5.5 nM T80896 C3JZH5 10183377 Ki = 15 nM T80896 CKT6Z4 10183386 IC50 = 266 nM T80896 CQB51M 10184149 IC50 = 24 nM T80896 C0J9AT 10184212 IC50 = 18.5 nM T80896 CG5N8H 10184413 Ki > 1000 nM T80896 C8XEP4 10192873 IC50 = 44 nM T80896 CR48FY 10192874 IC50 = 2933 nM T80896 CP70BT 10192899 IC50 = 1.5 nM T80896 C3RV4A 10192967 Ki = 18.9 nM T80896 CT19KI 10192968 Ki = 18.5 nM T80896 CVM71O 10192978 IC50 = 10 nM T80896 CY3ZU9 10193027 IC50 = 2.5 nM T80896 C1UF6W 10193573 IC50 = 150 nM T80896 C73GTR 10204098 IC50 = 300 nM T80896 CS91YM 10210142 Ki = 50 nM T80896 CH02FU 10214626 IC50 = 2 nM T80896 C4PKF0 10214678 Ki = 51 nM T80896 CJN2Y4 10214684 IC50 = 3200 nM T80896 CP90ZM 10214912 IC50 = 150 nM T80896 C82SVD 10215058 IC50 = 11 nM T80896 C8GZN0 10215089 IC50 = 1.7 nM T80896 CP4U5C 10215240 IC50 = 44 nM T80896 CP41MR 10215241 IC50 = 3 nM T80896 C7PSG6 10215290 IC50 = 0.5 nM T80896 C0FU1V 10215342 IC50 = 12 nM T80896 CP1S2V 10217796 IC50 = 115 nM T80896 CU2RI4 10217951 IC50 = 45 nM T80896 CW05OU 10218853 IC50 > 10000 nM T80896 CGF4E7 10226687 IC50 = 161 nM T80896 C7FXG9 10227720 IC50 = 223 nM T80896 C5M1RH 10229852 Ki = 30 nM T80896 CNB84J 10236378 IC50 = 42 nM T80896 CVMD95 10236407 IC50 = 1.2 nM T80896 CV9SZ3 10236450 IC50 = 6 nM T80896 C1K8OP 10236507 IC50 = 2 nM T80896 C7CPB9 10238739 IC50 = 20.3 nM T80896 CMY87N 10243978 EC50 = 0.37 nM T80896 C6RGH5 10244018 EC50 = 542 nM T80896 C7E0OP 10244111 IC50 = 27 nM T80896 CJQZ83 10254189 Ki = 0.9 nM T80896 CGV0O2 10268080 EC50 = 5 nM T80896 CPZY03 10275313 Ki = 8 nM T80896 C7LHP1 10275916 Ki = 630 nM T80896 CL5P3T 10276036 Ki = 190 nM T80896 CBD8V6 10282029 IC50 = 5 nM T80896 C7G4RE 10286186 IC50 = 13 nM T80896 C15UPR 10286213 IC50 = 1.1 nM T80896 C37GHD 10286369 IC50 = 3.4 nM T80896 C4U9ZV 10286370 IC50 = 10.6 nM T80896 CS4Y7Z 10286462 IC50 = 20 nM T80896 CM8IW0 10288944 IC50 = 64 nM T80896 CLOE40 10291224 IC50 = 103 nM T80896 C04JEC 10299557 IC50 = 5 nM T80896 C10CJA 10308134 IC50 = 2.3 nM T80896 CGR20A 10308169 IC50 = 2.4 nM T80896 C1KY6P 10308176 IC50 = 1.1 nM T80896 CX15KH 10308458 IC50 = 3.3 nM T80896 C7R4NE 10308501 Ki = 0.88 nM T80896 C0VUR6 10308538 IC50 = 150 nM T80896 COP14A 10312439 IC50 > 10000 nM T80896 COHA43 10316618 IC50 = 1.15 nM T80896 C0NX4P 10322799 IC50 = 45 nM T80896 C1FLQ0 10323601 Ki = 4 nM T80896 CPJS68 10324755 Ki = 4.19 nM T80896 C5K2CL 10332429 IC50 = 208 nM T80896 C7R6EP 10332721 IC50 = 82 nM T80896 CO2IH4 10334049 EC50 = 111 nM T80896 CPK7W1 10344612 Ki = 0.47 nM T80896 C0YAJ6 10344970 IC50 = 73 nM T80896 CEA16J 10344977 IC50 = 308 nM T80896 C7EF9B 10345685 IC50 = 9.1 nM T80896 C35BTN 10355544 IC50 = 10 nM T80896 CMY0N8 10355768 IC50 = 8 nM T80896 CL47OP 10356502 EC50 = 8506 nM T80896 C61WZX 10356510 IC50 = 69 nM T80896 C5YU0I 10358550 IC50 = 215 nM T80896 CR98BH 10358677 IC50 = 67 nM T80896 CKD8I0 10370518 IC50 = 111 nM T80896 CBG59N 10377168 IC50 = 75 nM T80896 CGCE89 10378417 IC50 = 14 nM T80896 CRB41T 10379126 EC50 = 8506 nM T80896 C6RQK1 10386584 IC50 > 10000 nM T80896 CK8MI6 10390296 IC50 = 52 nM T80896 CJV0O5 10400919 IC50 = 91 nM T80896 C7JN6F 10401620 IC50 = 22 nM T80896 C1P4XA 10414598 IC50 = 21.3 nM T80896 CA80YJ 10423234 EC50 = 76 nM T80896 C6H7EJ 10423780 IC50 = 35 nM T80896 CPM1L8 10425817 IC50 = 180 nM T80896 CC1V4Y 10428321 IC50 = 134 nM T80896 C98YGB 10430074 IC50 = 24 nM T80896 C8ZS3V 10447061 IC50 = 49.7 nM T80896 CZ08NR 10447944 IC50 = 99 nM T80896 CM92LK 10467580 IC50 = 54 nM T80896 C4JK0T 10468337 IC50 = 6.7 nM T80896 CLV49C 10470279 IC50 = 15.1 nM T80896 C6UMY7 10471178 IC50 = 44 nM T80896 CMG35I 10478373 IC50 = 31 nM T80896 C8GZN6 10479379 IC50 = 92.04 nM T80896 CHYB96 10480164 IC50 = 69 nM T80896 CZB0G1 10480448 Ki = 3.1 nM T80896 CM69RP 10768122 Ki = 35 nM T80896 C39FWK 10858337 EC50 = 21 nM T80896 CKTE95 10863480 Ki = 1800 nM T80896 CT1L6K 10874604 Ki > 10000 nM T80896 C2W9QX 10885394 IC50 = 2183 nM T80896 C75IVW 10892270 EC50 = 160 nM T80896 C4ZI0B 10897174 Ki = 790 nM T80896 CNZ9H2 10901682 EC50 = 257 nM T80896 CMW1U8 10906531 Ki = 820 nM T80896 CJP54O 10906754 Ki = 55 nM T80896 CY5R8D 10908233 Ki = 110 nM T80896 C40LHE 10917513 Ki > 10000 nM T80896 C3WI4P 10917876 IC50 = 492.04 nM T80896 CJ8OD1 10923143 EC50 = 35 nM T80896 CU46XG 10928571 IC50 = 421 nM T80896 CS24AP 10928882 IC50 = 396 nM T80896 COM46T 10929139 Ki = 15 nM T80896 CJ3RF6 10930298 Ki = 225 nM T80896 C3HG2S 10933614 EC50 = 120 nM T80896 C5E8VA 10938971 Ki = 3690 nM T80896 CK5D4I 10939453 IC50 = 47 nM T80896 CT8B7X 10940598 Ki = 40 nM T80896 C1OQB3 10945098 EC50 = 19000 nM T80896 CH14AY 10950078 Ki = 4200 nM T80896 CJL36T 10950356 Ki > 10000 nM T80896 CZ8F4V 10950649 IC50 = 105.93 nM T80896 CP2IK4 10950883 IC50 = 158.85 nM T80896 C3I5PB 10952341 Ki = 490 nM T80896 C4VD3H 10955612 EC50 = 1.4 nM T80896 CR94QD 10956181 EC50 = 302 nM T80896 CD90TL 10961334 Ki = 1000 nM T80896 CZGP46 10967017 EC50 = 1.7 nM T80896 CI9PC0 10972569 IC50 = 20 nM T80896 C7KSR9 10972765 Ki = 90 nM T80896 CW7ND8 10973721 Ki = 890 nM T80896 CW52ES 10973841 Ki = 115 nM T80896 CC4UT6 10978897 EC50 = 2 nM T80896 C93KBD 10978965 EC50 > 1000 nM T80896 CF2WJ3 10983822 Ki = 30 nM T80896 C2Q9UC 10985075 Ki = 425 nM T80896 C79JBL 10993930 IC50 = 82.99 nM T80896 CL1I0Z 10994057 Ki = 180 nM T80896 CW62AM 10999188 EC50 = 245 nM T80896 C1N8ZM 10999677 EC50 = 15 nM T80896 CGSE70 11011115 EC50 = 4.9 nM T80896 CE4C5I 11015765 IC50 = 198 nM T80896 CWO8S9 11016369 Ki = 170 nM T80896 CHR7A9 11016735 Ki = 25 nM T80896 CG37VC 11022432 EC50 = 186 nM T80896 CH9Y1B 11026647 IC50 = 33.04 nM T80896 CGX1N0 11028495 Ki = 110 nM T80896 CHM5C3 11030839 IC50 = 2400 nM T80896 COE9W8 11037182 Ki = 1750 nM T80896 CZW72E 11037591 IC50 = 354 nM T80896 C3JH4N 11039284 Ki = 200 nM T80896 CNG30Q 11048590 Ki = 4245 nM T80896 C2Z6TH 11048839 Ki = 490 nM T80896 CQN16G 11048858 IC50 = 302 nM T80896 C5W9IK 11060085 Ki = 105 nM T80896 CWO84P 11060104 Ki = 100 nM T80896 CV1A6F 11070590 Ki = 100 nM T80896 CF9LM6 11070635 Ki = 50 nM T80896 CU9PY6 11071460 Ki = 15 nM T80896 CWG41U 11075979 EC50 = 8 nM T80896 C2L7DT 11086416 EC50 = 249 nM T80896 C09ZLY 11088436 Ki > 10000 nM T80896 CG3VQ7 11091722 IC50 = 79.98 nM T80896 C8ED0O 11092497 Ki = 75 nM T80896 C49GHR 11097061 EC50 = 2.1 nM T80896 CX8YU9 11102748 IC50 = 1972.42 nM T80896 CD1G4U 11102972 Ki = 90 nM T80896 CR8OQ5 11114635 Ki = 400 nM T80896 CDJW25 11117751 EC50 = 69 nM T80896 C1O8RD 11124781 Ki = 600 nM T80896 CGH0S4 11135858 Ki = 100 nM T80896 CNEX86 11146178 Ki = 270 nM T80896 CJ4S8B 11153461 EC50 > 1000 nM T80896 CJ12UZ 11155391 IC50 = 13 nM T80896 CS2B4Z 11155392 IC50 = 39 nM T80896 CP7R9U 11156432 EC50 = 600 nM T80896 C4SEB7 11160528 EC50 = 5500 nM T80896 CGI4Y2 11162677 Ki = 375 nM T80896 CT0JD9 11164713 EC50 > 1000 nM T80896 C5DM4H 11165305 EC50 = 500 nM T80896 C68FNC 11167858 IC50 = 5950 nM T80896 CEML47 11172616 IC50 = 1100 nM T80896 CX91QE 11185437 IC50 = 10 nM T80896 CVAI71 11186162 IC50 = 128 nM T80896 CBS6E8 11197092 IC50 = 5.5 nM T80896 CAPL61 11197251 IC50 = 2.2 nM T80896 CLQ9C4 11197931 Ki = 0.44 nM T80896 C1XPD4 11201600 IC50 = 286 nM T80896 CB1FI6 11201991 IC50 = 19 nM T80896 C0M4IP 11208678 Ki = 6.92 nM T80896 CVK9E2 11214776 EC50 = 2800 nM T80896 C3M5WN 11224950 IC50 = 15 nM T80896 CA7F5T 11225110 EC50 = 3550 nM T80896 CN27ZJ 11231364 IC50 = 1.1 nM T80896 C2Q5PJ 11231792 IC50 = 6.9 nM T80896 C5IM4X 11247367 Ki = 0.19 nM T80896 C3RM9N 11254549 IC50 = 2.4 nM T80896 C5A7JR 11254851 IC50 = 6 nM T80896 CNJ4Q3 11255230 EC50 > 641 nM T80896 CYCR06 11256303 IC50 > 10000 nM T80896 CWF3M2 11256602 Ki = 0.7 nM T80896 CEA6U1 11259746 IC50 = 159 nM T80896 C7N9EL 11268331 IC50 = 4.5 nM T80896 C69KHE 11294796 IC50 = 19 nM T80896 C5A1NL 11300439 IC50 = 2.1 nM T80896 CS5HC9 11300885 EC50 = 5.3 nM T80896 CI7CZ3 11301461 IC50 = 2.6 nM T80896 C8S5AR 11314096 Ki = 0.41 nM T80896 C5M2KX 11317852 IC50 = 4.1 nM T80896 COU8G6 11323885 IC50 = 46 nM T80896 C1HZS7 11336351 IC50 > 10000 nM T80896 C1ZJ2R 11338969 IC50 = 496 nM T80896 CH12WB 11339036 IC50 = 879 nM T80896 CBN46V 11340868 Ki = 2.1 nM T80896 C2T7ZW 11350120 EC50 > 1000 nM T80896 CU6BE2 11350495 IC50 = 106 nM T80896 C6YUB4 11350836 IC50 = 173 nM T80896 CR1EB4 11351870 IC50 = 268 nM T80896 CSNT72 11357451 IC50 = 2 nM T80896 C8Z3YW 11359856 Ki = 0.46 nM T80896 CT3WZ0 11361524 IC50 = 464 nM T80896 C8AW4J 11363477 IC50 = 21 nM T80896 C90MRZ 11368962 EC50 = 38 nM T80896 C1HS3D 11369558 IC50 = 2.5 nM T80896 CMSU02 11370317 Ki = 10.2 nM T80896 C68GMX 11375318 EC50 = 470 nM T80896 CXO72T 11376166 EC50 = 400 nM T80896 CEI5V6 11385564 IC50 = 1945 nM T80896 CV98BT 11390181 IC50 = 10000 nM T80896 CK42BA 11391793 IC50 = 6.3 nM T80896 C8G2ED 11397112 IC50 = 238.8 nM T80896 C17SXG 11397412 IC50 = 29 nM T80896 CO15AK 11403179 IC50 = 1.2 nM T80896 CS6VA1 11406904 IC50 = 180 nM T80896 CUC6L8 11407390 IC50 = 162 nM T80896 CC9D7U 11427021 EC50 = 153 nM T80896 CM9VH4 11430588 IC50 = 252 nM T80896 CGF15N 11431657 IC50 = 276 nM T80896 C0VR7F 11437418 IC50 = 0.5 nM T80896 CP7J9V 11437506 IC50 = 3.4 nM T80896 C6QK5H 11441393 EC50 > 1000 nM T80896 C2NMY6 11465422 IC50 = 52 nM T80896 CFG6L2 11471499 IC50 = 7.3 nM T80896 C8B9ZT 11471500 IC50 = 4.4 nM T80896 CK75PT 11476995 IC50 = 11 nM T80896 CNUG46 11487991 IC50 = 143 nM T80896 C3PNE7 11493187 EC50 = 983 nM T80896 C7D5BU 11493338 IC50 = 3224 nM T80896 CFPW12 11496802 Ki = 0.5 nM T80896 CM76FT 11496925 Ki = 4.11 nM T80896 CQZ37A 11515143 EC50 = 9406 nM T80896 C4OBS2 11517134 Ki = 501 nM T80896 CJ2WY6 11522286 EC50 = 54 nM T80896 C9G5AE 11536973 IC50 = 25 nM T80896 C5W8HY 11537063 EC50 = 3.8 nM T80896 CMOL82 11540768 Ki = 1.16 nM T80896 C01NXW 11540918 EC50 = 1966 nM T80896 CW6KS5 11543706 EC50 = 750 nM T80896 CX7S6W 11551915 Ki = 421 nM T80896 CUK47O 11558075 EC50 = 2064 nM T80896 CWCZ35 11558237 EC50 = 62 nM T80896 CR4D8K 11558528 EC50 = 4.1 nM T80896 CP9GR8 11561520 Ki = 3 nM T80896 CUD60X 11565235 EC50 = 136 nM T80896 C5YO1V 11565733 EC50 = 1181 nM T80896 C7UDF3 11565847 IC50 = 7305 nM T80896 CFV87E 11565917 EC50 = 3843 nM T80896 C19NWZ 11565922 EC50 = 21 nM T80896 CWOZ42 11572578 EC50 = 9763 nM T80896 CPN71Y 11572694 EC50 = 7579 nM T80896 C26FJX 11582019 EC50 = 1638 nM T80896 C07ALM 11582925 Ki = 49.06 nM T80896 CKV64Z 11582975 Ki = 22 nM T80896 C4IZK8 11587711 EC50 = 37 nM T80896 CGM5O9 11589443 EC50 = 3804 nM T80896 C1FHL4 11594662 EC50 = 8776 nM T80896 C9QS7V 11605525 Ki = 54 nM T80896 CC21VD 11610867 Ki = 15 nM T80896 C3QV8F 11610940 EC50 = 593 nM T80896 CNP72K 11615788 EC50 = 0.3 nM T80896 CA3ID6 11619024 Ki = 48 nM T80896 CB10RY 11623915 EC50 = 8.7 nM T80896 C8M6GX 11631082 EC50 = 39 nM T80896 C7PG3I 11633183 Ki = 16 nM T80896 C45XNL 11637913 EC50 = 729 nM T80896 CQ8EI7 11638242 Ki = 2.2 nM T80896 C60DQS 11638602 EC50 = 68 nM T80896 CA7S2I 11644884 EC50 = 1254 nM T80896 C2MQE5 11644885 IC50 = 24 nM T80896 CD2TL1 11645057 EC50 = 52 nM T80896 C7NBT6 11645733 IC50 = 83 nM T80896 CK7ZQ8 11647673 IC50 = 2.1 nM T80896 C9LZ1F 11651922 EC50 = 904 nM T80896 CI1E3R 11659178 EC50 = 0.3 nM T80896 C3GXI8 11659260 EC50 = 117 nM T80896 C1QV8H 11660523 Ki = 118 nM T80896 C0LKN3 11663272 EC50 = 512 nM T80896 CF4HM7 11666535 EC50 = 1261 nM T80896 CX2W9Z 11666644 EC50 = 251 nM T80896 CJ2UC4 11674336 EC50 = 11685 nM T80896 CB1DU8 11674420 Ki = 0.49 nM T80896 C3IK0P 11680776 EC50 = 8870 nM T80896 CH7O4Y 11681405 IC50 = 249 nM T80896 CJL8A6 11681415 IC50 = 14 nM T80896 CFZ0K5 11688293 Ki = 2.8 nM T80896 CZ35CY 11694886 EC50 = 1313 nM T80896 COS65B 11695088 IC50 = 44265 nM T80896 CQ0IP3 11695307 IC50 = 48086 nM T80896 C20PTC 11696330 Ki = 0.91 nM T80896 CC6VK8 11702683 EC50 = 252 nM T80896 CG4E2O 11719093 Ki = 4 nM T80896 C43LND 11720175 Ki = 0.28 nM T80896 CRP5H6 11720774 Ki = 147 nM T80896 CR52IJ 11722356 EC50 = 379 nM T80896 C7D9HG 11724363 IC50 = 57 nM T80896 CO3S2Z 11724477 IC50 = 77 nM T80896 C4OH1Y 11726899 Ki > 10000 nM T80896 CWK56G 11730419 Ki = 170 nM T80896 CBMR23 11730420 Ki > 10000 nM T80896 C4FXP3 11730578 Ki = 20 nM T80896 C4GDB9 11730602 IC50 = 3687 nM T80896 CB8J4L 11730916 Ki = 15 nM T80896 C1I0ZW 11733031 Ki = 490 nM T80896 CT40UX 11734564 Ki = 210 nM T80896 CGZ40Y 11738040 IC50 = 5.6 nM T80896 C4DCI8 11738269 IC50 = 16 nM T80896 C9I3LZ 11738605 IC50 = 16 nM T80896 CCT71E 11743602 Ki = 200 nM T80896 C9KTN0 11744183 Ki = 4.9 nM T80896 C0K4LB 11749762 Ki > 1000000 nM T80896 CEC20W 11750375 IC50 = 287 nM T80896 C5YF3X 11750707 IC50 = 1155 nM T80896 C5JH1M 11751440 IC50 = 1370 nM T80896 CA2DO6 11770898 IC50 = 3 nM T80896 CHX6E0 11776977 IC50 = 310 nM T80896 CH7VT9 11777076 IC50 = 20 nM T80896 CD4W6C 11777154 IC50 = 67 nM T80896 C98FDE 11777375 EC50 = 13 nM T80896 CNLQ34 11777905 IC50 = 117 nM T80896 CT8OB2 11777956 EC50 = 358 nM T80896 CL76UG 11778912 IC50 = 28.1 nM T80896 CS9K7Z 11812018 IC50 = 82.99 nM T80896 C8YD5R 11823753 EC50 = 15 nM T80896 CYQ0W7 11826815 IC50 = 2202.93 nM T80896 CUVE20 11826959 Ki = 40 nM T80896 CT6Z4P 11827881 Ki = 40 nM T80896 C2VDT9 11954121 IC50 = 2200 nM T80896 CFB48H 11957006 IC50 = 12 nM T80896 C3F6JK 11977778 EC50 = 123 nM T80896 C2CXT4 11987846 IC50 = 1.5 nM T80896 CSK1Q4 12019124 IC50 > 5000 nM T80896 COR2Z7 12074176 Ki = 0.36 nM T80896 C2HNA8 12083341 IC50 = 127 nM T80896 COZ0Q5 12085941 IC50 = 93.3 nM T80896 C0P4TJ 12085942 IC50 = 2250 nM T80896 C41TJX 12258274 IC50 = 762 nM T80896 C5GV6L 13613337 IC50 = 218 nM T80896 C0BM7I 13868477 IC50 = 4000 nM T80896 CCF06L 15329708 IC50 = 1200 nM T80896 C42MYO 15429026 IC50 = 16.3 nM T80896 CB7K0N 15521393 IC50 = 260 nM T80896 CZ2F9Y 15541113 IC50 = 1800 nM T80896 C9IUR6 15543000 IC50 = 59 nM T80896 C0Q5RP 15543001 IC50 = 21 nM T80896 COW27A 15543007 IC50 = 37 nM T80896 CZB7P9 15543008 IC50 = 32 nM T80896 C8J6DM 15543009 IC50 = 9 nM T80896 CUO82C 15984114 EC50 = 0.4 nM T80896 C2CVH9 15984115 EC50 = 0.2 nM T80896 CWF0I6 16007239 EC50 = 5.5 nM T80896 CR2Q9N 16038396 Ki > 1000000 nM T80896 CV4LD2 16082545 IC50 > 1000 nM T80896 C7S4XY 16082546 IC50 = 1600 nM T80896 C5ZJR4 16082550 IC50 = 5800 nM T80896 CUOE19 16082557 IC50 = 180 nM T80896 CIWO01 16082558 IC50 = 100 nM T80896 CW2EC8 16082559 IC50 = 560 nM T80896 CZ3N1E 16082564 IC50 = 1200 nM T80896 C9WS2L 16082565 IC50 = 560 nM T80896 COR9P3 16082566 IC50 = 130 nM T80896 CH8A7C 16082568 IC50 > 10000 nM T80896 C9O5EM 16082572 IC50 = 510 nM T80896 CK7PI6 16082573 IC50 = 310 nM T80896 C9QXI4 16082574 IC50 = 230 nM T80896 C7GL5X 16082575 IC50 = 2200 nM T80896 C2BOE6 16103238 Ki = 192 nM T80896 C4UFW5 16103245 Ki = 156 nM T80896 C6H0EQ 16655080 IC50 = 1625 nM T80896 CU9LS2 16661702 IC50 > 10000 nM T80896 C1UY8J 16666386 IC50 > 5000 nM T80896 C1F5XE 16719760 IC50 = 2360 nM T80896 CE6FQ8 16719863 IC50 > 1600 nM T80896 C7N4LJ 16719865 Ki = 13.6 nM T80896 C0PMA8 16719866 IC50 = 48.6 nM T80896 CC82UX 16720250 IC50 = 66.7 nM T80896 CM4BS9 16739367 IC50 = 259 nM T80896 CZ34MS 16750039 IC50 = 1231 nM T80896 CVSA61 16750040 IC50 = 94 nM T80896 CQZK05 16758226 Ki = 0.53 nM T80896 CE4CP2 17756206 IC50 = 267 nM T80896 C4DV6C 17964485 Ki > 1000 nM T80896 C9B3MR 17972677 IC50 = 26 nM T80896 C4UG6E 17972712 IC50 = 69 nM T80896 CS1C5Q 18172400 IC50 = 48.8 nM T80896 C30ALH 18172403 IC50 = 22 nM T80896 CZ0VW4 18172409 IC50 = 63.5 nM T80896 C5U1YK 18172442 IC50 = 133 nM T80896 CJ05MC 18172444 IC50 = 180 nM T80896 CUS3Z9 18172448 IC50 = 27.9 nM T80896 C3X1FG 18172450 IC50 = 10.7 nM T80896 CTVK47 18172466 IC50 = 66.4 nM T80896 CR53UZ 18172469 IC50 = 71.2 nM T80896 C93MVX 18172476 IC50 = 220 nM T80896 CCE1L5 18172477 IC50 = 26.3 nM T80896 C0RZB8 18172482 IC50 = 27.4 nM T80896 C9DS4J 18695694 EC50 = 900 nM T80896 CGP29U 19793984 IC50 > 5000 nM T80896 C1F4KI 19793985 IC50 = 1980 nM T80896 C95KIE 20160413 IC50 = 140 nM T80896 CI0P6T 20161167 IC50 = 150 nM T80896 CM86ZJ 20734982 IC50 = 245 nM T80896 C0Q4FT 21051956 IC50 = 31 nM T80896 CF0S6J 21210483 IC50 = 23000 nM T80896 CV2N4Y 21252247 EC50 = 11 nM T80896 C7WBV5 21355678 IC50 = 8.9 nM T80896 CUL35V 21433016 IC50 = 180 nM T80896 C0HG2O 21625144 EC50 = 12 nM T80896 C6MTN2 21959300 IC50 = 77 nM T80896 CQS75R 22064611 Ki = 380 nM T80896 C89GZT 22221606 IC50 = 7.9 nM T80896 C5R3ZU 22221614 IC50 = 6.6 nM T80896 CD52LR 22221618 IC50 = 6 nM T80896 CU3E0Q 22221630 IC50 = 4 nM T80896 CN94JH 22221634 IC50 = 3.2 nM T80896 CC6X3H 22600576 IC50 > 10000 nM T80896 C6TJY8 23509070 EC50 = 1.1 nM T80896 C8FN7B 23648275 IC50 = 27.9 nM T80896 C4TNI0 23648457 Ki = 20.8 nM T80896 CZGS14 23648464 Ki = 0.26 nM T80896 CBL4I8 23648465 Ki = 0.745 nM T80896 CK0XL8 23648466 Ki = 5.97 nM T80896 C0GP7Q 23653178 EC50 = 4750 nM T80896 CV04HC 23653179 EC50 = 6890 nM T80896 CPR38W 24015539 EC50 = 1930 nM T80896 CTE1N2 24748569 EC50 > 10000 nM T80896 CP7M4B 24768258 EC50 > 1000 nM T80896 CH4QT2 24768259 EC50 > 1000 nM T80896 CC53XL 24860583 Ki > 2300 nM T80896 C2PGW1 24896626 IC50 = 9 nM T80896 CZC7L8 24953162 IC50 > 10000 nM T80896 C4W7BN 24954947 IC50 > 10000 nM T80896 C6XC2R 24954951 IC50 > 20000 nM T80896 CHY0D7 25013322 IC50 > 10000 nM T80896 C0TPS5 25013653 IC50 > 10000 nM T80896 CWU91M 25013811 IC50 > 10000 nM T80896 CSH29L 25013812 IC50 > 10000 nM T80896 C7J6IQ 25027904 EC50 = 9700 nM T80896 C4EGR5 25027907 IC50 = 220 nM T80896 CDK06N 25027908 IC50 = 83 nM T80896 CKY0G2 25028122 IC50 = 520 nM T80896 C0D3WT 25028125 IC50 = 2950 nM T80896 C4Z9PX 25028129 IC50 = 4900 nM T80896 CYVP87 25110671 IC50 = 2.9 nM T80896 CTYA32 25110672 IC50 = 0.7 nM T80896 CO41GX 25128805 Ki > 1000000 nM T80896 C4EI0A 25128806 Ki > 1000000 nM T80896 CQ34ZE 25128807 Ki > 1000000 nM T80896 CI19MZ 25128808 Ki > 1000000 nM T80896 COWS64 25128809 Ki > 1000000 nM T80896 C42RCW 25128810 Ki > 1000000 nM T80896 C8Q5ZK 25128811 Ki > 1000000 nM T80896 CD3Q4U 25128812 Ki > 1000000 nM T80896 C6V1ZT 25128813 Ki > 1000000 nM T80896 CAG08U 25128815 Ki > 1000000 nM T80896 C2FQX9 25128816 Ki > 1000000 nM T80896 C1HLM6 25129159 Ki > 1000000 nM T80896 C7QFR2 25129160 Ki > 1000000 nM T80896 C1PS3N 25129161 Ki > 1000000 nM T80896 CZS7Q1 25129163 Ki > 1000000 nM T80896 C1XZ5O 25129164 Ki > 1000000 nM T80896 C4YMG0 25129166 Ki > 1000000 nM T80896 CX70KG 25129167 Ki > 1000000 nM T80896 CGYS93 25129168 Ki > 1000000 nM T80896 C2E7NK 25129501 Ki > 1000000 nM T80896 CP7YX6 25129502 Ki > 1000000 nM T80896 CTX93Q 25129503 Ki > 1000000 nM T80896 CRA61L 25129504 Ki > 1000000 nM T80896 CV4AP7 25129505 Ki > 1000000 nM T80896 CZF6G7 25129855 Ki > 1000000 nM T80896 CNE47Z 25129856 Ki > 1000000 nM T80896 CC7FL0 25129857 Ki > 1000000 nM T80896 CV0W4X 25129858 Ki > 1000000 nM T80896 C6W5KP 25129859 Ki > 1000000 nM T80896 C9Z1YD 25129860 Ki > 1000000 nM T80896 CJ35NZ 25130215 Ki > 1000000 nM T80896 C2X5HD 25130216 Ki > 1000000 nM T80896 C94OVU 25130220 Ki > 1000000 nM T80896 C03ICO 25130561 Ki > 1000000 nM T80896 CZAN43 25130562 Ki > 1000000 nM T80896 C0IFU7 25130563 Ki > 1000000 nM T80896 CJT49R 25130564 Ki > 1000000 nM T80896 CRSM67 25130565 Ki > 1000000 nM T80896 CM8YT4 25130566 Ki > 1000000 nM T80896 CQ90UO 25130567 Ki > 1000000 nM T80896 COS0E1 25130893 Ki > 1000000 nM T80896 CR29KD 25130894 Ki > 1000000 nM T80896 CKX9J5 25130897 Ki > 1000000 nM T80896 CE9LJ6 25130898 Ki > 1000000 nM T80896 CV7WC6 25130899 Ki > 1000000 nM T80896 CJ4AK0 25130900 Ki > 1000000 nM T80896 C7HYX1 25131213 Ki > 1000000 nM T80896 C5PBM7 25131214 Ki > 1000000 nM T80896 C14WCP 25131215 Ki > 1000000 nM T80896 C7MVU3 25131217 Ki > 1000000 nM T80896 C1ZK7W 25131539 Ki > 1000000 nM T80896 CBGD76 25131540 Ki > 1000000 nM T80896 CX3NA8 25131542 Ki > 1000000 nM T80896 CX12DM 25131544 Ki > 1000000 nM T80896 CIQ2E4 25131893 IC50 > 1000000 nM T80896 C28UOB 25131894 Ki > 1000000 nM T80896 CK2ZT3 25131895 Ki > 1000000 nM T80896 CD13ZC 25131898 Ki = 132000 nM T80896 C1UZL6 25132248 Ki > 1000000 nM T80896 CIO06J 25132250 Ki > 1000000 nM T80896 CVFZ60 25132251 Ki > 1000000 nM T80896 CZX45O 25132598 Ki > 1000000 nM T80896 C2ANY3 25132599 Ki > 1000000 nM T80896 CC95RT 25132600 Ki > 1000000 nM T80896 C27KJG 25132602 Ki > 1000000 nM T80896 CQNY78 25132933 Ki = 2420 nM T80896 C6A8WM 25132934 Ki > 1000000 nM T80896 CO84WJ 25132935 Ki > 1000000 nM T80896 C6Z4IK 25132936 Ki > 1000000 nM T80896 C9JI7L 25132937 Ki > 1000000 nM T80896 CMYZ51 25132938 Ki > 1000000 nM T80896 CXO4C6 25132939 Ki > 1000000 nM T80896 C9DU6Q 25132940 Ki > 1000000 nM T80896 CZE3J7 25132941 Ki > 1000000 nM T80896 CR6ME8 25133259 Ki > 1000000 nM T80896 C0ET3J 25133260 Ki > 1000000 nM T80896 CK3VF4 25133261 Ki > 1000000 nM T80896 CB9K2T 25133267 Ki > 1000000 nM T80896 C6ZXQ0 25133268 Ki > 1000000 nM T80896 C9K0ZI 25133269 Ki > 1000000 nM T80896 C4RG8X 25133607 Ki > 1000000 nM T80896 CD3IH0 25133608 Ki > 1000000 nM T80896 CI82HF 25133609 Ki > 1000000 nM T80896 CM7VK8 25133611 Ki > 1000000 nM T80896 CD0NT6 25133612 Ki > 1000000 nM T80896 CWC8R0 25133614 Ki > 1000000 nM T80896 C2OCQ5 25133615 Ki > 1000000 nM T80896 CEC4P2 25133616 Ki > 1000000 nM T80896 CJ98GU 25133950 Ki > 1000000 nM T80896 C32UKW 25133951 Ki > 1000000 nM T80896 CE1WN2 25133952 Ki > 1000000 nM T80896 CNU20J 25133953 Ki > 1000000 nM T80896 C0V3KC 25133954 Ki > 1000000 nM T80896 CLT57Z 25133955 Ki > 1000000 nM T80896 CCW71Z 25133956 Ki > 1000000 nM T80896 CA76HY 25133959 Ki > 1000000 nM T80896 CI3RZ8 25133960 Ki > 1000000 nM T80896 C21XDY 25145083 Ki > 10000 nM T80896 CHDK07 25234182 EC50 = 46960 nM T80896 CLY9W3 25235364 IC50 > 10000 nM T80896 C3FW0Y 25257459 IC50 > 10000 nM T80896 CY6X2V 25258136 IC50 = 580 nM T80896 CV4Y6N 25258138 IC50 = 250 nM T80896 CLX0P9 25258381 IC50 > 10000 nM T80896 CNLS64 25258386 IC50 = 660 nM T80896 CSG7P9 25258611 IC50 = 3500 nM T80896 COM4U3 42609838 EC50 = 20000 nM T80896 C42TWL 44224340 EC50 = 170 nM T80896 C36BKU 44224542 EC50 = 1.1 nM T80896 C0FRP9 44224543 EC50 = 26 nM T80896 CEFT15 44224544 EC50 = 0.61 nM T80896 CLT65I 44225214 EC50 = 3.2 nM T80896 CS5PK0 44225454 EC50 = 8.4 nM T80896 CL1YK5 44225696 EC50 = 2.3 nM T80896 CFI64J 44227599 EC50 = 60 nM T80896 CXV83I 44227600 EC50 = 17 nM T80896 C40MCV 44275590 IC50 = 329 nM T80896 CY8L2T 44275591 IC50 = 103 nM T80896 CY1O5L 44280253 IC50 = 207 nM T80896 CHWV93 44280284 IC50 = 546 nM T80896 C3DS6O 44280299 IC50 = 598 nM T80896 CB32JI 44280300 IC50 = 1200 nM T80896 CP8D0O 44280322 IC50 = 1947 nM T80896 CFW6Y4 44280362 IC50 = 10000 nM T80896 CTB5L8 44280369 IC50 = 930 nM T80896 C2FE9I 44280602 IC50 > 10000 nM T80896 C5PKE0 44280604 IC50 = 5645 nM T80896 CD94FC 44280669 IC50 > 10000 nM T80896 C7SY2D 44280670 IC50 = 1200 nM T80896 C8YM6T 44280672 IC50 = 510 nM T80896 C6UQO3 44280673 IC50 = 152 nM T80896 CFG0A5 44280682 IC50 = 8.9 nM T80896 C9C6HY 44280687 IC50 = 7000 nM T80896 C8HK7P 44280689 IC50 > 10000 nM T80896 C0LNF3 44280705 IC50 = 454 nM T80896 CEX2O1 44280720 IC50 = 1360 nM T80896 CKUI19 44280721 IC50 = 1270 nM T80896 CPB4K1 44280724 IC50 = 5390 nM T80896 C9R3AO 44299445 Ki > 1000 nM T80896 CT2MK0 44299446 Ki = 65 nM T80896 C5B6IN 44300330 IC50 = 850 nM T80896 CP6A0S 44309223 IC50 = 70 nM T80896 CP52NB 44309415 IC50 = 183 nM T80896 CKG5Z0 44317015 IC50 = 1740 nM T80896 C2KD4V 44317238 IC50 = 343 nM T80896 CPKH32 44317395 IC50 = 1340 nM T80896 C2GZJ0 44317407 IC50 > 5000 nM T80896 CW21CA 44317747 Ki > 10000 nM T80896 C1HK7V 44319061 Ki = 0.06 nM T80896 CE9J8B 44319062 Ki = 0.91 nM T80896 C13KXZ 44319097 Ki = 0.43 nM T80896 CX6S1W 44319117 Ki = 20 nM T80896 C28JXF 44319637 IC50 = 105 nM T80896 C7S5JR 44319707 IC50 = 28 nM T80896 C58TKM 44319799 IC50 = 162 nM T80896 C7IXG8 44319951 IC50 = 40 nM T80896 C8GAE7 44319960 IC50 = 34 nM T80896 C4BID0 44319971 IC50 = 16 nM T80896 C4XTK5 44319973 IC50 = 43 nM T80896 CC5QD0 44319981 IC50 = 38 nM T80896 CXZP05 44320014 IC50 = 361 nM T80896 CIC5N6 44320017 IC50 = 8254 nM T80896 C7PS6E 44320029 IC50 = 60 nM T80896 CMLT05 44320030 IC50 = 8202 nM T80896 CRBN05 44325311 IC50 = 4.8 nM T80896 CD0IH3 44325322 IC50 = 1080 nM T80896 CNP05V 44325337 IC50 = 46.2 nM T80896 COTS43 44325352 IC50 = 41.7 nM T80896 C2B1OU 44325368 IC50 = 13.1 nM T80896 CZ9Y1O 44325433 IC50 > 3200 nM T80896 C5V7WZ 44325464 IC50 = 8.7 nM T80896 CS3R4P 44325467 IC50 = 295 nM T80896 C6NAY0 44325476 IC50 = 293 nM T80896 COL02R 44325510 IC50 = 185 nM T80896 CZ0P9W 44325539 IC50 = 595 nM T80896 CR94YN 44325546 IC50 = 788 nM T80896 C6TZA9 44325547 IC50 = 8 nM T80896 CML6J0 44325551 IC50 = 54 nM T80896 CL95JC 44325552 IC50 = 25 nM T80896 CDK3S0 44325556 IC50 = 13 nM T80896 CH8P0Z 44325557 IC50 = 520 nM T80896 C9DA8B 44325570 IC50 = 14 nM T80896 C6B7RO 44325581 IC50 = 13.2 nM T80896 C49BSH 44325582 IC50 = 73 nM T80896 CDX49O 44325585 IC50 = 413.2 nM T80896 CEAL30 44325586 IC50 = 105.4 nM T80896 CISM83 44325587 IC50 = 690 nM T80896 C8LG6M 44325589 IC50 = 1.1 nM T80896 C4K0RZ 44325613 IC50 = 7.3 nM T80896 CVD76C 44325614 IC50 = 792 nM T80896 CXYC85 44325632 IC50 = 350 nM T80896 CAE3Y9 44325639 IC50 = 109 nM T80896 C4S9ZI 44325650 IC50 = 67 nM T80896 CMJ0Z5 44325659 IC50 = 65.3 nM T80896 CEN5R9 44325692 IC50 = 18 nM T80896 C1SG7C 44348079 IC50 = 27 nM T80896 CSVW34 44348099 IC50 = 186 nM T80896 C1H7MO 44348132 IC50 = 27 nM T80896 CE4YL7 44348273 IC50 = 161 nM T80896 C28EVO 44348377 IC50 = 4372 nM T80896 C2GL8B 44348457 IC50 = 326 nM T80896 CXY05L 44348479 IC50 = 365 nM T80896 CWCS52 44348487 IC50 = 87 nM T80896 CQA68R 44348495 IC50 = 161 nM T80896 CE3O6Y 44348510 IC50 = 583 nM T80896 C0I9FH 44348522 IC50 = 186 nM T80896 CLX35U 44348531 IC50 = 115 nM T80896 CX82TV 44348539 IC50 = 59 nM T80896 C90INV 44348540 IC50 = 259 nM T80896 C3B6LK 44355916 EC50 = 0.15 nM T80896 CK1UW9 44355917 EC50 = 0.14 nM T80896 CBO3X2 44355927 EC50 = 30 nM T80896 CIWX06 44356135 EC50 = 110 nM T80896 CW67AN 44356136 EC50 = 0.41 nM T80896 CM7H1I 44356536 EC50 = 3.7 nM T80896 C7UH6W 44356621 Ki = 17 nM T80896 CYBO90 44356823 Ki = 120 nM T80896 C4UTM7 44356833 Ki = 73 nM T80896 CT07FI 44389476 EC50 = 183 nM T80896 CG80UZ 44389487 EC50 = 25 nM T80896 CL92HF 44389493 EC50 = 24 nM T80896 COW1E9 44389558 EC50 = 3.1 nM T80896 C5ECY2 44389569 EC50 = 79 nM T80896 CY5K2O 44389570 EC50 = 275 nM T80896 CRN5I1 44389572 EC50 = 318 nM T80896 CL7C9P 44389577 EC50 = 3164 nM T80896 CZJ5C4 44389581 EC50 = 9.2 nM T80896 C9Q4UB 44389582 EC50 = 6 nM T80896 CSP4T9 44389593 EC50 = 305 nM T80896 CEHT06 44389595 EC50 = 7.2 nM T80896 CTJ9Q6 44389606 EC50 = 2825 nM T80896 CS47PF 44389609 EC50 = 25 nM T80896 CUA5F4 44389617 EC50 = 197 nM T80896 CVT09Q 44389633 EC50 = 485 nM T80896 CV24GJ 44389648 EC50 = 3050 nM T80896 C8MI1L 44389650 EC50 = 39 nM T80896 C9RUX6 44389654 EC50 = 67 nM T80896 CL2W9P 44389655 EC50 = 6 nM T80896 CQ01VW 44389659 EC50 = 12 nM T80896 C2PDC8 44389876 IC50 = 25.29 nM T80896 C8ZIP3 44389878 IC50 = 3.21 nM T80896 CA05VL 44389880 IC50 = 66.52 nM T80896 CB1H3E 44389883 IC50 = 19.77 nM T80896 CUP57N 44389890 IC50 = 93.57 nM T80896 CBIA52 44389891 IC50 = 1.27 nM T80896 CQU8C6 44389896 IC50 = 20.09 nM T80896 C10LSB 44389901 IC50 = 7.92 nM T80896 C6CIB9 44389904 IC50 = 29.37 nM T80896 C8YNX2 44389906 IC50 = 9.07 nM T80896 C39DPH 44389907 IC50 = 12.9 nM T80896 C2ZS9G 44389914 IC50 = 4.94 nM T80896 C19MKQ 44389919 IC50 = 17.67 nM T80896 C4W5VU 44389922 IC50 = 14.22 nM T80896 CB7K5Y 44389934 IC50 = 3.7 nM T80896 CVG41F 44389943 IC50 = 12.47 nM T80896 CO1H5G 44389945 IC50 = 18.15 nM T80896 C8GD3V 44389948 IC50 = 4.02 nM T80896 CP0Y8G 44390069 IC50 = 4.5 nM T80896 C1JQD2 44390070 IC50 = 627 nM T80896 CPFB84 44390071 IC50 = 18 nM T80896 C24ZDP 44390072 IC50 = 11 nM T80896 CXHL23 44390084 IC50 = 171 nM T80896 CQ92BW 44390097 IC50 = 26 nM T80896 C6RC2Y 44390116 IC50 = 179 nM T80896 C4GP0U 44390120 IC50 = 23 nM T80896 C1DS5R 44390163 IC50 = 16 nM T80896 C7ZQ1J 44391057 IC50 = 315 nM T80896 C50XAP 44391076 IC50 = 110 nM T80896 C5Y6CT 44391206 IC50 = 3.6 nM T80896 C0ZIT7 44391782 IC50 = 13 nM T80896 CS4XD9 44391788 IC50 = 363 nM T80896 CV4G0H 44391842 IC50 = 44 nM T80896 CRJE53 44391854 IC50 = 13 nM T80896 C5W2IH 44391860 IC50 = 176 nM T80896 CZOJ29 44391870 IC50 = 15 nM T80896 CIT5P8 44391879 IC50 = 81 nM T80896 C0B5IT 44391881 IC50 = 46 nM T80896 CZH85I 44391888 IC50 = 114 nM T80896 CQD42M 44391889 IC50 = 59 nM T80896 CT0BO6 44391890 IC50 = 97 nM T80896 C1NIS3 44391905 IC50 = 38 nM T80896 C74EHI 44391917 IC50 = 25 nM T80896 C7RVQ5 44391988 IC50 = 90 nM T80896 CP15SF 44392410 IC50 = 3111.72 nM T80896 CA82NU 44392580 IC50 = 10 nM T80896 CC72ZY 44392593 IC50 = 3.3 nM T80896 CDMN93 44392636 IC50 = 0.35 nM T80896 CS8ZN5 44393200 IC50 = 39 nM T80896 CP53NK 44393219 IC50 = 85 nM T80896 CB5DS4 44393237 IC50 = 33 nM T80896 C1GA9N 44393240 IC50 = 81 nM T80896 C0TLH5 44393249 IC50 = 366 nM T80896 CL27NW 44393263 IC50 = 18 nM T80896 CR64AD 44393267 IC50 = 59 nM T80896 CTN81R 44393286 IC50 = 118 nM T80896 CW59RL 44393287 IC50 = 116 nM T80896 C01ODV 44393310 IC50 = 47 nM T80896 C82WUF 44393322 IC50 = 247 nM T80896 CO1Q0W 44393335 IC50 = 51 nM T80896 C0JXU4 44393336 IC50 = 72 nM T80896 CC89WN 44393340 IC50 = 26 nM T80896 C2WXI0 44393342 IC50 = 81 nM T80896 CNP73S 44393366 IC50 = 33 nM T80896 C8E0AJ 44393367 IC50 = 436 nM T80896 CQY82B 44393380 IC50 = 40 nM T80896 CP25CW 44393381 IC50 = 331 nM T80896 C8P3FU 44393399 IC50 = 52 nM T80896 CIS79C 44393400 IC50 = 267 nM T80896 C1XOK4 44393405 IC50 = 56 nM T80896 CV5YB6 44393408 IC50 = 1113 nM T80896 CRB41V 44393419 IC50 = 275 nM T80896 C5U2KP 44394160 IC50 = 2 nM T80896 C13SYV 44396250 Ki = 39 nM T80896 CB1P0S 44396251 Ki = 13 nM T80896 CHY1C3 44396271 Ki = 240 nM T80896 C29MBI 44396272 Ki = 160 nM T80896 C4TQ6N 44396282 Ki = 89 nM T80896 CH2Y3L 44396283 Ki = 13 nM T80896 CWZB52 44396284 Ki = 190 nM T80896 CD80LM 44396296 Ki = 570 nM T80896 C6SI5L 44396297 Ki > 750 nM T80896 C45LRH 44396317 Ki = 30 nM T80896 C5JG6H 44396330 Ki = 48 nM T80896 CA8V4G 44396331 Ki > 750 nM T80896 CD2EY3 44399091 IC50 = 1150 nM T80896 CDJ7H0 44399199 IC50 = 199 nM T80896 CK1X0O 44400690 IC50 = 28 nM T80896 CSE07P 44402388 IC50 = 7.26 nM T80896 CSZ2J0 44402418 IC50 = 16.4 nM T80896 C6I3PD 44402432 IC50 = 53.9 nM T80896 C3FR5B 44402483 IC50 = 31 nM T80896 C6CWQ3 44402516 IC50 = 21.4 nM T80896 CC3QK6 44402532 IC50 = 25 nM T80896 CM35QL 44402545 IC50 = 16.6 nM T80896 CL9CQ8 44402598 IC50 = 45.6 nM T80896 CN57AQ 44402634 IC50 = 215 nM T80896 CQH5B1 44402654 IC50 = 20.2 nM T80896 CF0VN8 44402705 IC50 = 35 nM T80896 C7VCZ5 44402711 IC50 > 10000 nM T80896 CXI97U 44402746 IC50 > 10000 nM T80896 CGRX27 44402769 IC50 > 10000 nM T80896 C9XS4E 44402799 IC50 > 10000 nM T80896 CB2V0A 44403942 Ki = 3.8 nM T80896 CARV69 44405133 IC50 = 0.9 nM T80896 CKZ15D 44405150 IC50 = 0.6 nM T80896 CR4V3M 44405163 IC50 = 3.1 nM T80896 C2C9OW 44405166 IC50 = 2.6 nM T80896 CG85OU 44405167 IC50 = 2.4 nM T80896 CLE8X1 44405174 IC50 = 2.3 nM T80896 C72SFE 44405903 IC50 = 149 nM T80896 C79JEI 44407631 EC50 = 8 nM T80896 CB0L6S 44407636 EC50 = 171 nM T80896 C2W0PF 44407655 IC50 = 1619 nM T80896 CWU1O4 44407658 IC50 = 132 nM T80896 C6J3VA 44407760 EC50 = 188 nM T80896 C1O6WJ 44407763 EC50 = 827 nM T80896 C21CBM 44407771 EC50 = 78 nM T80896 CD3E0R 44407782 EC50 = 96 nM T80896 C2O1DA 44407785 EC50 = 67 nM T80896 CXD31Y 44407857 EC50 = 379 nM T80896 C4K3ZG 44408764 IC50 = 13 nM T80896 C7CSE3 44408771 IC50 = 2340 nM T80896 CF06GJ 44408808 IC50 = 19 nM T80896 C1K3FC 44409005 IC50 = 7.8 nM T80896 C5HM2W 44409078 IC50 = 26 nM T80896 CIUR71 44409233 IC50 = 957 nM T80896 CC7O0B 44409614 EC50 = 11342 nM T80896 CF0IQ7 44412807 IC50 = 4220 nM T80896 CI4KN9 44412821 IC50 = 123 nM T80896 C5E9XO 44412823 IC50 = 32 nM T80896 C5S9OV 44412835 IC50 = 945 nM T80896 CN9X6E 44412848 IC50 > 10000 nM T80896 CE60QX 44412849 IC50 = 15 nM T80896 CZ13IC 44412903 IC50 = 2.5 nM T80896 C3ADY8 44412904 IC50 = 16 nM T80896 CJ4S8E 44412954 IC50 = 936 nM T80896 C0JAX2 44412955 IC50 = 374 nM T80896 C4EZB6 44412956 IC50 = 4.5 nM T80896 CW08IO 44412979 IC50 = 188 nM T80896 CFH31O 44412983 IC50 = 4.4 nM T80896 C5RT0I 44413033 IC50 = 19 nM T80896 C2TFX6 44413049 IC50 = 1810 nM T80896 CE2P7W 44413050 IC50 = 313 nM T80896 CQW1N9 44414035 EC50 = 0.8 nM T80896 CXBZ80 44414036 EC50 = 0.8 nM T80896 C2H8RD 44414046 IC50 = 1.1 nM T80896 CQC9F4 44414050 EC50 = 210 nM T80896 CIS2L0 44414060 EC50 = 1.5 nM T80896 CJBQ27 44414066 EC50 = 0.9 nM T80896 C09CRE 44414068 IC50 = 8 nM T80896 CECT78 44414069 IC50 = 5.2 nM T80896 CI12OU 44414094 EC50 = 0.6 nM T80896 CF5T6Y 44414110 IC50 = 0.8 nM T80896 CGP27O 44414111 EC50 = 5.8 nM T80896 CXG13L 44414126 EC50 = 2.1 nM T80896 C8E5PN 44414131 EC50 = 0.7 nM T80896 CV1LR4 44414182 IC50 = 4 nM T80896 CALJ60 44414245 IC50 = 0.3 nM T80896 C5WTR2 44414246 IC50 = 1 nM T80896 C7MT9J 44414260 IC50 = 4.1 nM T80896 CL0K4C 44414274 IC50 = 0.9 nM T80896 C90LXU 44414284 EC50 = 935 nM T80896 C0I3YZ 44414292 IC50 = 7 nM T80896 CPFS03 44414293 IC50 = 1.1 nM T80896 C7L2PW 44415352 IC50 = 28 nM T80896 C2Y9BF 44415353 IC50 = 14 nM T80896 C96JSR 44415397 IC50 > 10000 nM T80896 C5V2SP 44415478 IC50 = 1 nM T80896 C7YQ9X 44415498 IC50 = 11 nM T80896 CREK89 44415499 IC50 = 5 nM T80896 C18JCA 44415511 IC50 = 45 nM T80896 CGS79I 44415523 IC50 = 5 nM T80896 C1FCL0 44415547 IC50 = 141 nM T80896 C6PD3R 44415553 EC50 = 2.3 nM T80896 CH50DC 44415571 EC50 = 0.96 nM T80896 CSF5O8 44415669 EC50 = 4.9 nM T80896 C7C4XF 44415699 EC50 = 28 nM T80896 CCO34X 44415700 EC50 = 0.4 nM T80896 C3KI0H 44415761 IC50 = 1524 nM T80896 CV37CW 44415788 EC50 = 5.8 nM T80896 CG72WC 44427370 Ki = 1.69 nM T80896 C2F8CW 44427371 Ki = 2.17 nM T80896 CHB94D 44427372 Ki = 0.35 nM T80896 CYB7J6 44427373 Ki = 0.16 nM T80896 CQ96LY 44427374 Ki = 0.29 nM T80896 CN2M3P 44427375 Ki = 2.69 nM T80896 CQ74SE 44427404 Ki = 0.63 nM T80896 CHK6A4 44427405 Ki = 15.7 nM T80896 CL1Y4N 44430357 IC50 > 5000 nM T80896 C5S6XP 44430360 IC50 > 5000 nM T80896 CUQT28 44430361 IC50 > 5000 nM T80896 CKF6I1 44430362 IC50 > 5000 nM T80896 COT67E 44430364 IC50 = 2810 nM T80896 C2YF4G 44430366 IC50 = 560 nM T80896 CBGX08 44430369 IC50 > 5000 nM T80896 CY4XR5 44430372 IC50 = 92 nM T80896 C27KUN 44430374 IC50 = 2810 nM T80896 C6LV9A 44430376 IC50 = 339 nM T80896 CHM5G2 44430378 IC50 > 5000 nM T80896 CJ5G2Z 44439806 IC50 = 4900 nM T80896 CG17VZ 44439807 IC50 = 78 nM T80896 C5Y4CM 44439809 IC50 = 1582 nM T80896 C28PCX 44439811 IC50 > 10000 nM T80896 C4WS3E 44439813 IC50 > 10000 nM T80896 C3H6BA 44439815 IC50 > 10000 nM T80896 C3DGB7 44439820 IC50 = 5594 nM T80896 CL9IE2 44439822 IC50 = 2954 nM T80896 C7RLX5 44439823 IC50 = 2340 nM T80896 C1A0PH 44439825 IC50 = 394 nM T80896 C3KS9O 44439826 IC50 = 4749 nM T80896 CFZ0N1 44439827 IC50 = 2653 nM T80896 CMW5Z8 44439828 IC50 > 10000 nM T80896 CWBD12 44439829 IC50 = 3250 nM T80896 C2Y4GR 44439830 IC50 = 3688 nM T80896 CZNS72 44439831 IC50 = 2338 nM T80896 COGW71 44439832 IC50 = 606 nM T80896 C76TMP 44439833 IC50 = 2236 nM T80896 C82NQD 44439834 IC50 = 426 nM T80896 C98BPO 44439835 IC50 = 161 nM T80896 C1HZ2K 44439836 IC50 = 522 nM T80896 C3LO1U 44440237 EC50 = 4 nM T80896 CLK05T 44440238 IC50 = 16 nM T80896 CP3JU8 44440239 IC50 = 3020 nM T80896 C34ERB 44440240 EC50 = 132 nM T80896 C5KG7L 44440241 EC50 = 219 nM T80896 CB1ZS3 44440262 EC50 = 28 nM T80896 CKON02 44440263 EC50 = 198 nM T80896 C5DB8N 44440264 EC50 = 440 nM T80896 C89JEW 44440265 EC50 > 1000 nM T80896 CR7G2K 44440266 EC50 > 1000 nM T80896 CVT4O9 44440267 EC50 > 1000 nM T80896 CO98DZ 44440268 EC50 > 1000 nM T80896 CC73BF 44440269 EC50 = 86 nM T80896 CL3WI5 44441857 EC50 = 240 nM T80896 CIL2C9 44441858 EC50 > 1000 nM T80896 CR2S3A 44441859 IC50 = 115 nM T80896 C6GRK9 44441860 EC50 > 1000 nM T80896 C2FC5N 44441861 EC50 = 170 nM T80896 CA1BY2 44441862 EC50 = 480 nM T80896 C6SMB2 44441863 EC50 = 31 nM T80896 CTQ15A 44441864 EC50 = 190 nM T80896 CF06VH 44441865 EC50 = 24 nM T80896 C1X5MS 44441866 IC50 = 120 nM T80896 CNQ96S 44450617 IC50 = 2900 nM T80896 C2BCU6 44450633 IC50 = 2100 nM T80896 CYG7X4 44473146 IC50 > 10000 nM T80896 CT0B2Q 44473422 EC50 > 1000 nM T80896 CR5SI0 44476535 EC50 > 10000 nM T80896 CM29JD 44516036 IC50 > 10000 nM T80896 C3ND5A 44542643 EC50 > 1000 nM T80896 C3SBL5 44543099 EC50 > 1000 nM T80896 C8DNR7 44566760 EC50 = 19 nM T80896 CEI26D 44569027 Ki > 1000000 nM T80896 CCPW27 44569028 Ki > 1000000 nM T80896 CF4RS6 44569029 Ki > 1000000 nM T80896 CEA0U9 44579680 Ki = 30 nM T80896 C8W6ZF 44580025 Ki = 170 nM T80896 CXGP15 44580026 Ki = 110 nM T80896 CW5O3K 44580027 Ki = 162 nM T80896 CZOU20 44589952 IC50 = 46.1 nM T80896 CNM79D 44589953 IC50 = 5.9 nM T80896 C1JCM3 44589998 IC50 = 4.61 nM T80896 CDP6W8 44589999 IC50 = 3.63 nM T80896 C5FC9V 44590000 IC50 = 31 nM T80896 CYI29S 44590098 IC50 = 6 nM T80896 CD8R7Y 44590099 IC50 = 262 nM T80896 C7T8KP 44590100 IC50 > 15000 nM T80896 C4RZX5 44590136 IC50 = 8.78 nM T80896 C6NZW2 44590137 IC50 = 17.33 nM T80896 CL7IT6 44592556 IC50 = 2048 nM T80896 C4VM3B 44592558 IC50 = 15030 nM T80896 CKYW84 44596355 IC50 = 31 nM T80896 CY0U6X 44596356 IC50 = 380 nM T80896 CQG0F7 44596357 IC50 > 1000 nM T80896 CSR28W 44596358 IC50 > 1000 nM T80896 CAG36H 44596359 IC50 = 105 nM T80896 C6AZU3 44596467 IC50 = 108 nM T80896 C49XRU 44596468 IC50 = 125 nM T80896 C1YRA4 44596469 IC50 = 99 nM T80896 CS12MF 44596470 IC50 = 108 nM T80896 C2K1DR 44596471 IC50 = 66 nM T80896 C3LMA0 44596573 IC50 = 205 nM T80896 C3KH5Y 44596574 IC50 = 140 nM T80896 CJM37H 44596575 IC50 = 200 nM T80896 C8GJ9B 44596686 IC50 = 16 nM T80896 CSQ10X 44596687 IC50 = 200 nM T80896 CFJE97 44596688 IC50 = 23 nM T80896 CYX0C2 44596789 IC50 = 30 nM T80896 CM67OY 44596790 IC50 = 24 nM T80896 CUT7N3 44596791 IC50 = 63 nM T80896 CAI8D6 44596792 IC50 > 10000 nM T80896 C9KW4Y 44596793 IC50 = 12 nM T80896 CBLN03 44596894 IC50 > 1000 nM T80896 CX76YZ 44596895 IC50 = 28 nM T80896 CLWY41 44596896 IC50 = 41 nM T80896 CSUT20 44596897 IC50 = 18.5 nM T80896 CRUO49 44596898 IC50 > 1000 nM T80896 C1FI6O 44596992 IC50 = 22 nM T80896 C0YUC1 44596993 IC50 = 63 nM T80896 CN1M3J 44596994 IC50 = 13.4 nM T80896 C6NEV4 44596995 IC50 = 24 nM T80896 C42NEY 44596996 IC50 = 8.7 nM T80896 CUK16W 44597094 IC50 = 11 nM T80896 C43LCQ 44597095 IC50 = 11 nM T80896 CLJM84 44597096 IC50 = 31 nM T80896 C9R2CP 44597097 IC50 = 390 nM T80896 CL01OK 44597098 IC50 = 580 nM T80896 CMR68J 44597209 IC50 = 18.6 nM T80896 CWG9Z7 44597210 IC50 = 5.68 nM T80896 CYA0B6 44597211 IC50 = 44 nM T80896 CE31LY 44597212 IC50 = 19 nM T80896 C9QO1F 44597743 IC50 = 23 nM T80896 C63LWP 44597744 IC50 = 20 nM T80896 C3O2NE 44597745 IC50 = 19 nM T80896 CME14J 44597857 IC50 = 14 nM T80896 CI9E7J 44597858 IC50 = 35 nM T80896 C95YGF 44597859 IC50 = 27 nM T80896 CD9EL6 44597860 IC50 = 86 nM T80896 C6GWQ8 44597861 IC50 = 0.64 nM T80896 CS79YT 44597968 IC50 = 12.7 nM T80896 CUO92A 44597969 IC50 = 11 nM T80896 CMXI54 44597970 IC50 = 44 nM T80896 CT9Q0J 44597971 IC50 = 16 nM T80896 CSOD50 44597973 IC50 = 250 nM T80896 CIJP09 44605898 IC50 > 10000 nM T80896 C08UBE 45272032 IC50 > 10000 nM T80896 C5C8ZD 46237712 EC50 = 174 nM T80896 CP1VU0 46237713 EC50 = 221.31 nM T80896 C0HMU5 46237838 EC50 = 34.59 nM T80896 C6RZX9 46237839 EC50 = 22.65 nM T80896 CKBD82 46237840 EC50 = 242.1 nM T80896 CPD64X 46237841 EC50 = 26.67 nM T80896 CL6SY4 46866497 IC50 = 22000 nM T80896 CO1T3Q 46871902 IC50 = 41700 nM T80896 C9UZ5N 46871916 IC50 = 96000 nM T80896 CDHA57 46880834 IC50 > 30000 nM T80896 CN9L7G 46916268 IC50 = 550 nM T80896 C05YMH 46935020 EC50 = 150 nM T80896 CX0NO8 49782554 EC50 < 12531.41 nM T80896 CC7T8Q 49782555 EC50 < 15240.53 nM T80896 CD07EV 49782777 EC50 < 8336.81 nM T80896 C43UKW 49782778 EC50 = 5188 nM T80896 C2JTF0 49782779 EC50 = 52 nM T80896 CS7KX9 49782780 EC50 = 2398.83 nM T80896 C36RYU 49782781 IC50 < 4045.76 nM T80896 C8OA0C 49782985 EC50 < 2747.89 nM T80896 C5Y6QU 49782986 EC50 = 129.42 nM T80896 CB8V7R 49782987 EC50 < 19364.22 nM T80896 CUD91T 49862248 EC50 = 534000 nM T80896 C0SY6G 49864608 EC50 = 0.07 nM T80896 C2JAP4 50919273 EC50 = 3800 nM T80896 C0BPT6 50919274 EC50 = 310 nM T80896 CY10IC 50940834 EC50 = 251.19 nM T80896 CTH45Q 52918523 IC50 > 10000 nM T80896 CF16DR 52937206 EC50 = 227000 nM T80896 CG7LY6 52937207 EC50 = 1600 nM T80896 CS0UY6 52937307 EC50 = 3200 nM T80896 CB94DP 52937308 EC50 = 60000 nM T80896 C75SPY 52937309 EC50 = 30000 nM T80896 C80AYX 52937310 EC50 = 1000 nM T80896 CYA61L 53323081 IC50 = 63 nM T80896 CWHK62 53483961 EC50 = 79 nM T80896 C5ZX4B 54597874 IC50 > 10000 nM T80896 C8GP2M 56658858 EC50 = 14 nM T80896 C0HMP7 56662184 EC50 = 43 nM T80896 CRTW04 56662185 EC50 > 2400 nM T80896 CH65JX 56662340 EC50 = 101 nM T80896 C1WS4G 56662341 EC50 = 65 nM T80896 CWY30K 56665645 EC50 > 3000 nM T80896 CFQ51I 56672695 EC50 = 51 nM T80896 C9CXS4 56675930 EC50 = 1100 nM T80896 CZT8H6 56676055 EC50 = 84 nM T80896 C9ZJ8I 56679386 EC50 = 110 nM T80896 CP06XK 56679387 EC50 = 48 nM T80896 CP58AC 56679388 EC50 = 1480 nM T80896 CK1N6F 56682681 EC50 = 418 nM T80896 CG8J9I 56682682 EC50 = 437 nM T80896 C53OZE 56945585 EC50 = 0.76 nM T80896 C37IJX 57392620 IC50 = 6.8 nM T80896 CTM6K5 57690900 IC50 > 5000 nM T80896 C87TXE 57992044 EC50 = 11 nM T80896 CI6XF5 58742295 IC50 > 3200 nM T80896 CYI71B 58902727 EC50 = 66 nM T80896 CE18JH 60202715 EC50 = 35.2 nM T80896 C2F5TS 68037237 EC50 = 27.5 nM T80896 C16MVN 68058524 EC50 = 1400 nM T80896 CMT2I3 68321354 IC50 = 1300 nM T80896 C7KM0T 68779769 IC50 = 13 nM T80896 CBM80I 70354859 EC50 = 35.2 nM T80896 C4NMI7 70681450 IC50 = 3.1 nM T80896 CID9L6 70681451 IC50 = 2.6 nM T80896 C6YL4K 70681621 EC50 = 160 nM T80896 CARO49 70685018 Ki = 51 nM T80896 CLO8E7 70690044 EC50 = 760 nM T80896 C1KFL5 70690047 EC50 = 1870 nM T80896 CWGC38 70692196 EC50 = 4400 nM T80896 CY7EL2 70694264 EC50 = 1270 nM T80896 CP5QM9 70696352 EC50 = 14000 nM T80896 C4PIS1 71153303 IC50 = 2.512 nM T80896 CK61DU 71296056 EC50 = 6600 nM T80896 CG24SA 71449116 IC50 = 5.53 nM T80896 COPG39 71454424 EC50 = 220 nM T80896 CYW34A 71519686 IC50 = 2700 nM T80896 CT9Y5D 71549558 IC50 = 2400 nM T80896 C8ZX0F 71549573 IC50 = 15000 nM T80896 CZ8Y7O 71549829 IC50 = 5300 nM T80896 CPFL57 71549843 IC50 = 15000 nM T80896 CY8SP0 71549969 IC50 = 7300 nM T80896 CX6JR5 71550242 IC50 = 2700 nM T80896 C6WIA2 71550244 IC50 = 2600 nM T80896 CPL0O7 71624342 EC50 = 1940 nM T80896 C9S4KZ 71624466 EC50 = 610 nM T80896 CA7F2B 71624467 EC50 = 1920 nM T80896 CGT86N 71624573 EC50 = 780 nM T80896 C1RV0Q 71624574 EC50 = 203 nM T80896 C2CLE1 71624678 EC50 = 1340 nM T80896 CD23NV 71624679 EC50 = 660 nM T80896 COK59Y 71624683 EC50 = 5700 nM T80896 CN06AS 71624796 EC50 = 1230 nM T80896 CFW3R0 71624797 EC50 = 2460 nM T80896 CT1KP7 71624798 EC50 = 10800 nM T80896 C5Y9LF 71624799 EC50 = 295 nM T80896 C2C0LQ 71624915 EC50 = 2230 nM T80896 C1PD9I 71625173 EC50 = 5110 nM T80896 C5XEQ9 71625175 EC50 = 17500 nM T80896 C0OY8P 71661130 EC50 = 49210 nM T80896 CM3N9E 71712303 IC50 = 380 nM T80896 CNRU01 71712304 IC50 = 43 nM T80896 C8EY6K 71714518 IC50 = 2600 nM T80896 CLM0A3 71714519 IC50 = 4500 nM T80896 C5NU0T 71721539 IC50 = 15200 nM T80896 CGJ5X4 71812208 IC50 = 200 nM T80896 CN9M7E 71817803 EC50 = 12 nM T80896 CI20JH 72188710 EC50 = 33800 nM T80896 CW36SK 73057389 IC50 = 6.8 nM T80896 CIS0D4 73057390 IC50 = 9.8 nM T80896 CP0Y4U 73057391 IC50 = 88 nM T80896 CJQ93L 73057392 IC50 = 108 nM T80896 C7WEA2 73057393 IC50 = 111 nM T80896 C1AUC0 73057394 EC50 = 99 nM T80896 C5AUY4 73347354 EC50 = 72400 nM T80896 CK3RU8 73347518 IC50 = 800 nM T80896 C4XOW1 73348859 EC50 = 17690 nM T80896 CXL50F 73350442 EC50 = 25300 nM T80896 CY53FM 73351956 EC50 = 4280 nM T80896 CQN6M8 73353409 EC50 = 4680 nM T80896 C0G1IK 73353410 EC50 = 2760 nM T80896 C9WY3B 73386689 EC50 = 9.5 nM T80896 CP5E2V 76333018 EC50 = 125.89 nM T80896 C9CL2H 76335717 IC50 > 25000 nM T80896 CA0D6H 76336630 EC50 = 0.3981 nM T80896 C1B5KS 76336631 EC50 = 19.95 nM T80896 C5JK1L 89042295 EC50 = 11 nM T80896 CK5D1A 90395281 IC50 = 12000 nM T80896 C1J2TA 90654352 IC50 = 804 nM T80896 C4BA8W 90656430 IC50 = 34800 nM T80896 CA9PL8 91663316 IC50 = 10400 nM T80896 CNJH98 102502192 EC50 = 18 nM T80896 C5ZR2C 102502193 EC50 = 28 nM T80896 C17BIZ 118097387 EC50 = 680 nM T80896 CI4GP9 118097391 EC50 = 42 nM T80896 C6NIU0 118724546 IC50 = 56000 nM T80896 C3JU5H 118724548 IC50 = 980 nM T80896 C4UB8J 118724549 IC50 = 4800 nM T80896 CE0C6J 118724550 IC50 = 1200 nM T80896 C7BRJ0 118724551 IC50 = 1100 nM T80896 C5LR2N 118724552 IC50 = 19 nM T80896 CG1OL3 118724553 IC50 = 23000 nM T80896 CCK94J 118724554 IC50 = 144000 nM T80896 CW07TL 118724555 IC50 = 15 nM T80896 COJ81W 118735362 EC50 = 49.2 nM T80896 C8VFT2 118735363 EC50 = 202 nM T80896 CZE92I 118735364 EC50 = 182 nM T80896 CFB1G7 118735365 EC50 = 49.9 nM T80896 CX4V1E 118735366 EC50 = 19.5 nM T80896 CW60ZD 118735367 EC50 = 27.8 nM T80896 C6ULM1 118735368 EC50 = 52 nM T80896 CE50LC 118735369 EC50 = 36.5 nM T80896 C6Y2NQ 118735371 EC50 = 478 nM T80896 C93CNO 118735374 EC50 = 519 nM T80896 C4YR6E 118735375 EC50 = 47.7 nM T80896 CS3ZJ8 118735376 EC50 = 57.5 nM T80896 CV83KA 118735377 EC50 = 1350 nM T80896 CG9RB4 118735379 EC50 = 21.3 nM T80896 CGT60X 118735380 EC50 = 13.3 nM T80896 CY6L8W 118735381 EC50 = 293 nM T80896 CG13LX 122178361 IC50 = 3000 nM T80896 CRW9F3 122180812 IC50 = 330 nM T80896 C3UO8M 122180813 Ki = 1416.67 nM T80896 CJ42OQ 122180814 IC50 = 160 nM T80896 CRH37W 122180815 Ki = 629.63 nM T80896 CEW23B 122180816 Ki = 126.87 nM T80896 CBM0N2 122180817 Ki = 653.85 nM T80896 C7E2QD 122180818 Ki = 87.32 nM T80896 CBO5T8 122180819 Ki = 67.73 nM T80896 C3TB4Y 122180820 Ki = 618.18 nM T80896 C3D4TV 122180821 Ki = 81.53 nM T80896 CC80JD 122180822 Ki = 91.89 nM T80896 CXPG14 122180823 Ki = 101.49 nM T80896 CS4OH2 122180824 Ki = 39.04 nM T80896 CB7MD5 122180825 Ki = 95.24 nM T80896 CB51GT 122180826 Ki = 49.78 nM T80896 C1YZ6A 122180827 Ki = 121.43 nM T80896 CYCT17 122180828 Ki = 200.01 nM T80896 COM0C9 122180829 Ki = 60.5 nM T80896 CP5ND8 122180830 Ki = 255.64 nM T80896 CTPJ86 122180831 Ki = 478.87 nM T80896 C4FJ1W 122180832 Ki = 971.43 nM T80896 CF71OE 122180833 IC50 = 89 nM T80896 CL16JS 122180834 Ki = 55.65 nM T80896 CE2A5S 122180835 EC50 = 2 nM T80896 CBC6D3 122181041 EC50 = 38 nM T80896 CP4ZJ2 122181042 EC50 = 54 nM T80896 COEZ74 122181043 EC50 = 203 nM T80896 C0EHV1 122181044 EC50 = 23 nM T80896 CA0KZ7 122181045 EC50 = 2 nM T80896 CE4AO3 122181046 EC50 = 173 nM T80896 C7XP2A 122181047 Ki = 809.52 nM T80896 CYD03G 122181048 Ki = 102.41 nM T80896 CD6M1W 122190205 EC50 = 45840 nM T80896 C10SKD 122190207 EC50 = 5650 nM T80896 C4P9NG 122700657 EC50 = 24 nM T80896 CZPJ13 122700846 EC50 = 6290 nM T80896 CB5WZ1 122702036 EC50 = 1570 nM T80896 C6CA4O 124088406 EC50 = 33 nM T80896 CNH4A8 124088429 EC50 = 75 nM T80896 C4M8QN 127030254 IC50 = 40 nM T80896 C3QCS2 127033894 IC50 = 260 nM T80896 CZS07N 127049269 IC50 = 155 nM T80896 C4ITS1 127050198 IC50 = 1660 nM T80896 C2REL0 127051417 IC50 = 41 nM T80896 CBF64U 127051803 IC50 = 190 nM T80896 C12WOQ 129137247 EC50 = 70.8 nM T80896 CJB4M3 129137266 EC50 = 857 nM T80896 CJ1N2M 129137280 EC50 = 486.2 nM T80896 CH42QX 129137285 EC50 = 1263 nM T80896 CK1BE9 134155077 EC50 = 346.4 nM T80896 C2BK3Z 134155779 EC50 = 218.4 nM T80896 C67KRX 135348923 EC50 = 250 nM T80896 CT70RL 135348926 EC50 = 2700 nM T80896 CU87GS 135348929 EC50 = 21000 nM T80896 C1G9FD 135348960 EC50 = 49 nM T80896 C42PVJ 135400902 IC50 = 5 nM T80896 CL51KF 135400937 IC50 = 17 nM T80896 CBRN70 135400938 IC50 = 2 nM T80896 CY2GJ3 135401184 IC50 = 192 nM T80896 CLX32H 135409570 Ki = 122 nM T80896 C6S5RV 135409748 IC50 = 5.3 nM T80896 CY39LP 135409961 IC50 = 79 nM T80896 CO95DR 135409966 IC50 = 3.7 nM T80896 CMQE75 135412817 IC50 = 12 nM T80896 C1VWL3 135415992 IC50 = 190 nM T80896 CPC1Q3 135421346 Ki = 25.12 nM T80896 CLN16H 135423261 IC50 = 1.4 nM T80896 C3BU7D 135423323 Ki = 10 nM T80896 CCRX48 135424620 IC50 = 3 nM T80896 CP9JN3 135424801 EC50 = 173 nM T80896 C0KIP8 135425149 EC50 = 222 nM T80896 CXNV83 135430308 IC50 = 6 nM T80896 C30QWY 135430315 IC50 = 28 nM T80896 CK2ZF0 135431815 IC50 = 1040 nM T80896 CYJ7R0 135432882 IC50 = 2.4 nM T80896 CWCV13 135433141 Ki = 1410 nM T80896 CA1MC6 135433906 IC50 = 1.8 nM T80896 CW7MZ8 135436561 IC50 = 356 nM T80896 CAY0S9 135436566 IC50 = 750 nM T80896 CCR8P7 135438141 IC50 = 37 nM T80896 CC29NQ 135438201 IC50 = 112 nM T80896 CDA4B8 135438473 EC50 = 53 nM T80896 CUXH34 135440385 Ki = 25.12 nM T80896 CBGO63 135443283 IC50 = 32 nM T80896 C8VWH0 135443287 IC50 = 1600 nM T80896 CX1T4W 135443301 IC50 = 42 nM T80896 C21VTE 135445165 Ki = 63.1 nM T80896 C5M9IX 135445349 IC50 = 1340 nM T80896 CE50DW 135445365 IC50 = 102 nM T80896 C60OGT 135445374 IC50 = 366 nM T80896 CVM0P7 135446139 EC50 = 160 nM T80896 CTD6A7 135449071 IC50 = 33 nM T80896 C9GZ1Q 135454811 IC50 = 211 nM T80896 CEQ5F4 135457031 IC50 > 5000 nM T80896 C9BVI8 135457325 IC50 = 3 nM T80896 C2O1MP 135457889 Ki = 48 nM T80896 C1Z4BN 135458008 IC50 = 3.6 nM T80896 CCVE26 135458128 IC50 = 27 nM T80896 CXU79B 135458129 IC50 = 221 nM T80896 CY8U6E 135459005 IC50 > 100000 nM T80896 CHU54B 135461939 IC50 = 95 nM T80896 CEB1W8 135471179 IC50 > 5000 nM T80896 CPO9D1 135477943 IC50 = 3.4 nM T80896 C17LIP 135481146 IC50 = 26 nM T80896 C4O7RZ 135481158 IC50 = 201 nM T80896 C8SE4C 135483639 IC50 = 40 nM T80896 C6V1JZ 135483640 IC50 = 1 nM T80896 C6DI2R 135483660 IC50 = 25 nM T80896 C0WP9D 135486163 EC50 = 4.3 nM T80896 CH9OV8 135487481 EC50 = 20 nM T80896 CFO4V6 135489088 IC50 = 23 nM T80896 CQ91HA 135489089 IC50 = 44 nM T80896 CAU4W8 135489212 Ki = 630.96 nM T80896 CXY1Z2 135492323 IC50 = 31 nM T80896 CMB9Z7 135493223 IC50 = 64 nM T80896 CTN2D6 135495080 IC50 = 1.9 nM T80896 CX3O9M 135495087 IC50 = 66 nM T80896 CFDO01 135496191 IC50 = 166 nM T80896 CB9Q3X 135496242 Ki = 15.85 nM T80896 CMK68Q 135497123 IC50 = 155 nM T80896 C90ZNW 135497128 Ki = 19.95 nM T80896 C2O8MY 135499764 IC50 = 96 nM T80896 CI09WX 135499787 IC50 = 93 nM T80896 CE1D4V 135499837 IC50 = 52 nM T80896 C25GWU 135500024 IC50 = 87 nM T80896 CRYW41 135502641 IC50 = 14 nM T80896 C1RW9U 135503521 IC50 = 4.4 nM T80896 COF53G 135507181 Ki = 680 nM T80896 CPZ29O 135508382 IC50 = 6 nM T80896 C2ME7Q 135508383 IC50 = 135 nM T80896 C9GM1V 135508397 IC50 = 313 nM T80896 CFMN96 135511852 EC50 = 7 nM T80896 C7PZI5 135511869 EC50 = 13 nM T80896 C61NSW 135514474 Ki = 251.19 nM T80896 CV6B8P 135515561 Ki = 110 nM T80896 C4XD9K 135516685 IC50 = 20 nM T80896 CGM5C6 135516694 IC50 = 1.5 nM T80896 CZKC69 135518123 IC50 = 20 nM T80896 CBPO32 135518124 IC50 = 879 nM T80896 CVTD54 135518270 IC50 = 36 nM T80896 C3S5MX 135518313 IC50 = 64 nM T80896 CH6G0Q 135519304 IC50 = 138 nM T80896 C3P8LZ 135519309 IC50 = 12 nM T80896 CU5J8M 135520120 IC50 = 440553 nM T80896 CR03JM 135522279 IC50 = 59 nM T80896 C1OBI2 135524469 IC50 = 25 nM T80896 CVX9H3 135524526 IC50 = 3.1 nM T80896 CMIE65 135524868 IC50 > 5000 nM T80896 C7TYU2 135524871 IC50 = 97 nM T80896 CC46RN 135524945 Ki = 1584.89 nM T80896 CFQW27 135526994 IC50 = 10 nM T80896 CSZ1H7 135527005 EC50 = 47 nM T80896 CRKD27 135529495 Ki = 710 nM T80896 CQ0ZX7 135529496 Ki > 3000 nM T80896 CX1J8D 135535917 IC50 = 8 nM T80896 C15FTQ 135538030 IC50 = 2.4 nM T80896 CUCN57 135540445 IC50 = 27 nM T80896 CIKD94 135545359 IC50 = 2.2 nM T80896 C7X2CE 135547714 IC50 = 40 nM T80896 CK7UM1 135547715 Ki = 178 nM T80896 C34JMK 135571931 IC50 > 100000 nM T80896 C4ODC2 135678114 Ki = 1515 nM T80896 CDJ1L6 135914665 EC50 = 37500 nM T80896 CMJ41H 135987657 Ki = 1050 nM T80896 CO0UC2 135987660 Ki = 1170 nM T80896 CP96SU 135987662 Ki = 660 nM T80896 C3I8VE 135987663 Ki = 1100 nM T80896 CDG17Y 135987664 Ki > 3000 nM T80896 C9ABZ6 135987665 Ki = 250 nM T80896 C7GU8Q 135987666 Ki = 1000 nM T80896 C4G1DL 135987668 Ki = 790 nM T80896 CIG6T5 135987670 Ki = 1120 nM T80896 C1TV3R 135987671 Ki = 1260 nM T80896 CSB76X 135987672 Ki = 330 nM T80896 C98FXW 136046127 IC50 = 13 nM T80896 CUN8F1 136046128 IC50 = 6 nM T80896 CX2KM3 136046129 IC50 = 41 nM T80896 CFQ9U2 136046130 IC50 = 45 nM T80896 CSOR78 136046131 IC50 = 19 nM T80896 CB1L2D 136046132 IC50 = 16 nM T80896 CQTA24 136046133 IC50 = 9 nM T80896 CB6YN3 136046134 IC50 = 24 nM T80896 CJ7AO4 136046135 IC50 = 7 nM T80896 C68OIK 136046136 IC50 = 6 nM T80896 CQ7K2A 136046137 EC50 = 332 nM T80896 CSCP10 136046138 EC50 = 628 nM T80896 C2CL1K 136046139 EC50 = 2 nM T80896 C9LMN8 136046140 IC50 = 51 nM T80896 CJSU38 136046141 EC50 = 10860 nM T80896 CU18VS 136046142 IC50 = 6 nM T80896 C5ORA9 136046143 IC50 = 67 nM T80896 CFGU03 136046144 IC50 = 180 nM T80896 CJ8X1O 136046145 IC50 = 28 nM T80896 C4P2BT 136046146 IC50 = 139 nM T80896 CXTR87 136046147 IC50 = 100 nM T80896 C9BI5M 136046148 IC50 = 417 nM T80896 CAH5S3 136046149 EC50 = 276 nM T80896 C0YZM4 136048726 IC50 = 3.2 nM T80896 CMI3Z2 136048727 IC50 = 16 nM T80896 C1BE8P 136048728 IC50 = 23 nM T80896 CRVT63 136048730 IC50 = 45 nM T80896 CZG20O 136053633 EC50 = 30 nM T80896 CJC8N5 136053634 EC50 = 160 nM T80896 CV3TP6 136053635 EC50 = 120 nM T80896 CNW6H0 136053636 EC50 = 18 nM T80896 C5WTV7 136053637 EC50 = 26 nM T80896 CRBK35 136053638 EC50 = 8 nM T80896 CRV6U5 136053639 EC50 = 16 nM T80896 C54YLG 136053640 EC50 = 240 nM T80896 CCB5P6 136053641 EC50 = 270 nM T80896 CO60LF 136053642 EC50 = 180 nM T80896 CB54HV 136053643 EC50 = 77 nM T80896 CRA6C4 136053644 EC50 = 140 nM T80896 C2MB8E 136099749 IC50 = 166 nM T80896 CC1UT0 136099750 IC50 = 1.4 nM T80896 C4F5VO 136099751 IC50 = 3.2 nM T80896 C36UFX 136099752 IC50 = 142 nM T80896 C4MW6I 136099753 IC50 = 45 nM T80896 CL1ZT0 136099754 IC50 = 16 nM T80896 C9ZHF5 136099755 IC50 = 313 nM T80896 CM35UY 136180341 EC50 = 3.97 nM T80896 CXP07U 136180342 EC50 = 14.7 nM T80896 C94TFC 137287868 EC50 = 225 nM T80896 C56DIS 137349270 IC50 = 0.631 nM T80896 CM7X1H 137637325 EC50 = 207 nM T80896 C2N3FX 137638822 IC50 = 2525 nM T80896 CLTS71 137641590 IC50 = 154 nM T80896 CRS0C8 137643006 IC50 = 306 nM T80896 CL9W7S 137648342 EC50 = 343 nM T80896 C8FVM1 137649725 EC50 = 894 nM T80896 CMR9Z4 137652975 IC50 = 939 nM T80896 C1AS5K 137653286 IC50 = 1690 nM T80896 CUPZ80 137657526 IC50 = 1977 nM T80896 CM3UF7 137700779 IC50 > 20000 nM T80896 CCF02H 145964530 IC50 = 10000 nM T80896 C56SHA 145964597 IC50 = 5900 nM T80896 CMG6W2 145964616 EC50 = 63 nM T80896 CVJ7L6 145964633 Ki = 226.37 nM T80896 C8QI0U 145965134 Ki = 12.8 nM T80896 C5H8EZ 145965425 IC50 = 7400 nM T80896 CM9LG0 145965903 Ki = 115.08 nM T80896 C8K1WV 145965925 EC50 = 43 nM T80896 CA6CZ4 145966389 EC50 = 194 nM T80896 CS9MD6 145966668 Ki = 167.48 nM T80896 C0WG5H 145966819 Ki = 722.81 nM T80896 CE4S7F 145967279 EC50 = 3 nM T80896 CNJO46 145967622 IC50 = 354 nM T80896 C80AGW 145967704 IC50 = 175 nM T80896 CB68HI 145967819 IC50 = 14340 nM T80896 C8KNI7 145967847 IC50 = 1014 nM T80896 C8H3YV 145968201 IC50 = 0.55 nM T80896 C1S0TJ 145968278 IC50 = 3.1 nM T80896 CXN86W 145968289 IC50 = 43 nM T80896 CE1WK0 145968307 IC50 = 34 nM T80896 C8BF1J 145968369 IC50 = 0.94 nM T80896 CRUO57 145968523 IC50 = 1.23 nM T80896 C2CE4P 145968537 IC50 = 447 nM T80896 CD86FU 145968562 IC50 = 585 nM T80896 CT8R7I 145968943 EC50 = 941 nM T80896 CY0VA4 145969440 IC50 = 25 nM T80896 CO75XN 145969585 IC50 = 72 nM T80896 CEY2I5 145969791 IC50 = 46 nM T80896 C7PQH3 145969854 Ki = 59.71 nM T80896 CXY0E1 145970107 IC50 = 72 nM T80896 CVW6D7 145972047 Ki = 321.88 nM T80896 C4KJX2 145972317 EC50 = 749 nM T80896 CDQ7E0 145972963 EC50 = 5760 nM T80896 C4OF2V 145973074 EC50 = 276 nM T80896 C37FBS 145973441 EC50 = 139 nM T80896 C3AZ4O 145973866 Ki = 50 nM T80896 CXZS64 145974009 EC50 = 242 nM T80896 CQZ7D8 145975059 EC50 = 31 nM T80896 CE5N1B 145976228 Ki = 180.7 nM T80896 C4Q9KI 145976280 Ki = 528.21 nM T80896 C8DS5Q 145976853 EC50 = 2 nM T80896 C4DPO7 145976892 EC50 = 4 nM T80896 CRJU43 145976968 EC50 = 9 nM T80896 CO70FX 145977155 Ki > 10000 nM T80896 C7IL3R 145977161 IC50 = 69 nM T80896 CVX45W 145977605 Ki = 179.91 nM T80896 C9MG6O 145977673 Ki = 121.53 nM T80896 C98CHS 145977976 IC50 = 23600 nM T80896 C43SYL 145978903 IC50 = 475 nM T80896 C1AJL5 145979357 IC50 = 5 nM T80896 CCBN24 145979638 IC50 = 299 nM T80896 CJ3R5P 145980235 EC50 = 509 nM T80896 CE80KP 145980527 EC50 = 240 nM T80896 CJ5U0Y 145980901 IC50 = 1120 nM T80896 CLJ3S7 145981530 IC50 = 16 nM T80896 CVC58M 145981549 IC50 = 2960 nM T80896 C21SIT 145981553 IC50 = 540 nM T80896 CSM61H 145981867 EC50 = 1147 nM T80896 CCRI70 145983336 Ki = 390 nM T80896 CP27UK 145983884 Ki = 77 nM T80896 CYZO43 145984038 Ki = 25 nM T80896 CVJY47 145984216 Ki = 1.2 nM T80896 CO50ZW 145985605 Ki = 3640 nM T80896 C3O4HE 145985821 Ki = 64 nM T80896 CN91YC 145986320 IC50 = 1335 nM T80896 CMQK52 145986591 IC50 = 119 nM T80896 C28LAH 145986759 IC50 = 1159 nM T80896 CA1D2B 145987043 IC50 = 203 nM T80896 CPRH38 145987084 IC50 = 102 nM T80896 CF9S0O 145987265 IC50 = 395 nM T80896 CKYW98 145988223 IC50 = 1945 nM T80896 CK5RV0 145988666 EC50 = 600 nM T80896 C09MNB 145988825 IC50 = 2.4 nM T80896 C7I9CZ 145989448 EC50 = 435 nM T80896 CW0C8Y 145989462 IC50 = 5391 nM T80896 CX74YQ 145989561 EC50 = 51 nM T80896 CSF03L 145989681 IC50 = 1235 nM T80896 CR0LK9 145989755 IC50 = 415 nM T80896 COI2R8 145991129 IC50 = 1266 nM T80896 C2NH3M 145991296 IC50 = 331 nM T80896 CP4V8N 145991796 IC50 = 43 nM T80896 CLR23U 155519218 IC50 = 3000 nM T80896 CNU6O4 155525430 EC50 = 1.2 nM T80896 C4ID8Q 155539669 IC50 = 1300 nM T80896 C31CNR 155541121 IC50 = 1500 nM T80896 CP9Y8J 155548583 IC50 = 2700 nM T80896 C5MHU4 155552943 IC50 = 1400 nM T80896 CY28HU 155567231 IC50 > 5000 nM T80896 C4JTH2 155568868 IC50 = 180 nM T80896 C0RGJ9 44389594 EC50 = 1.4 nM T80896 D00CWN 135987619 Ki = 35 nM T80896 D00DJX 44597742 IC50 = 21 nM T80896 D00HZT 135449109 IC50 = 533 nM T80896 D00IXB 10445833 IC50 = 3.2 nM T80896 D00NEK 44405867 IC50 = 355 nM T80896 D00RIX 5280443 IC50 = 130 nM T80896 D00URP 10399473 IC50 = 74 nM T80896 D00ZBL 135458122 IC50 = 13 nM T80896 D01AHL 44412953 IC50 = 1530 nM T80896 D01CYI 11579721 EC50 = 961 nM T80896 D01GPY 10192794 IC50 = 10 nM T80896 D01IAT 10171410 IC50 = 566 nM T80896 D01KJU 6102690 IC50 = 2.52 nM T80896 D01KSR 135495079 IC50 = 157 nM T80896 D01QXL 9993627 IC50 = 15 nM T80896 D01SWO 9901869 IC50 = 28 nM T80896 D01TUB 135519319 IC50 = 4.6 nM T80896 D01WCA 656936 IC50 = 6 nM T80896 D02DML 5281707 IC50 = 2 nM T80896 D02EJM 136048731 IC50 = 1.42 nM T80896 D02GLM 9994500 Ki = 2800 nM T80896 D02HGS 135502634 IC50 = 30 nM T80896 D02JJU 135492380 IC50 = 521 nM T80896 D02LCC 135442595 IC50 = 82 nM T80896 D02OKF 10308197 IC50 = 1.4 nM T80896 D02RQP 6623 EC50 = 1100 nM T80896 D02TPO 10323679 IC50 = 7 nM T80896 D02WIL 7433743 Ki > 10000 nM T80896 D02WRU 11201035 Ki = 139 nM T80896 D02WSA 11579722 EC50 = 1721 nM T80896 D02XVV 10399376 IC50 = 93 nM T80896 D03BOO 25128804 Ki > 1000000 nM T80896 D03CBX 135454802 IC50 = 4.3 nM T80896 D03DVM 10131379 IC50 = 12 nM T80896 D03GYS 135499774 IC50 = 79 nM T80896 D03QHG 16066665 IC50 = 141 nM T80896 D03RYU 135522275 IC50 = 3 nM T80896 D03XEU 10286022 IC50 = 10 nM T80896 D04EAY 135474202 IC50 = 254 nM T80896 D04SAO 9799518 IC50 = 3 nM T80896 D04TPC 25130896 IC50 > 1000000 nM T80896 D04WHH 135519317 IC50 = 11 nM T80896 D05EOW 102614 EC50 = 0.71 nM T80896 D05FUY 10149584 IC50 = 9 nM T80896 D05GKC 108003 EC50 = 38 nM T80896 D05JKC 135546593 IC50 = 16 nM T80896 D05JPW 135409725 IC50 = 59 nM T80896 D05KXP 44418726 IC50 = 421 nM T80896 D05LQD 10082995 IC50 = 326 nM T80896 D05PNP 11064571 IC50 = 14700 nM T80896 D05YIU 10236250 IC50 = 1.6 nM T80896 D06DDT 5315502 EC50 = 530 nM T80896 D06OAL 135442585 IC50 = 13 nM T80896 D06SCS 135418373 IC50 = 1.4 nM T80896 D07HBQ 25128814 Ki = 299000 nM T80896 D07LUI 11459006 IC50 = 16 nM T80896 D07VPM 135409756 IC50 = 235 nM T80896 D07XBD 10308075 IC50 = 17 nM T80896 D07XUY 44418717 IC50 = 863 nM T80896 D08FLV 135474625 IC50 = 46 nM T80896 D08HCF 135496133 IC50 = 703 nM T80896 D08SJL 135524856 IC50 = 75 nM T80896 D08VDX 10214699 IC50 = 2.3 nM T80896 D08WDN 135496123 IC50 = 718 nM T80896 D09CQC 135471161 IC50 = 50 nM T80896 D09DEK 10171409 IC50 = 44 nM T80896 D09FWP 11368353 IC50 = 2000 nM T80896 D09FWS 135430317 IC50 = 52 nM T80896 D09NOH 44418728 IC50 = 59 nM T80896 D09PXU 9991961 IC50 = 88 nM T80896 D09TQE 135528620 IC50 = 66 nM T80896 D09UWI 14905189 EC50 = 1540 nM T80896 D0AD3U 135528621 IC50 = 39 nM T80896 D0AU0M 637542 EC50 = 4890 nM T80896 D0B1HP 135526958 IC50 = 54 nM T80896 D0C5FY 10331951 IC50 = 46 nM T80896 D0C6AP 10285954 IC50 = 5.6 nM T80896 D0C9XK 135545334 IC50 = 105 nM T80896 D0C9XW 11276767 Ki = 16000 nM T80896 D0CC6R 10125290 IC50 = 2 nM T80896 D0D1LB 44418733 IC50 = 244 nM T80896 D0DK9S 135454786 IC50 = 3660 nM T80896 D0F1SS 44605900 IC50 > 3000 nM T80896 D0FD6Z 10308090 IC50 = 1.6 nM T80896 D0H1CO 10244394 IC50 = 1050 nM T80896 D0H2FI 10308268 IC50 = 199 nM T80896 D0H5HI 9993278 IC50 = 45 nM T80896 D0H6MZ 25133613 Ki > 1000000 nM T80896 D0H8PI 10308021 IC50 = 5.8 nM T80896 D0HM8Y 44408971 IC50 = 49 nM T80896 D0HR8L 11447703 IC50 = 205 nM T80896 D0I5HZ 44405888 IC50 = 137 nM T80896 D0I5VJ 135520257 EC50 = 14 nM T80896 D0J0AG 135421237 IC50 = 88 nM T80896 D0J2NG 44418724 IC50 = 69 nM T80896 D0K0IC 13896065 IC50 = 1.12 nM T80896 D0K0TR 11356877 IC50 = 680 nM T80896 D0K1TW 135443280 IC50 = 239 nM T80896 D0K6TE 10286087 IC50 = 11 nM T80896 D0K7HR 135409729 IC50 = 60 nM T80896 D0K8QD 63059 EC50 = 306.9 nM T80896 D0L2MU 10286352 IC50 = 2 nM T80896 D0L3AX 236868 IC50 = 245 nM T80896 D0L6IQ 135424609 IC50 = 1190 nM T80896 D0LI0M 44418723 IC50 = 97 nM T80896 D0M0XL 11414445 IC50 = 114 nM T80896 D0MY8V 10308207 IC50 = 8.4 nM T80896 D0N0OY 135405741 IC50 = 49 nM T80896 D0NN0V 637048 IC50 = 880 nM T80896 D0O2KP 12133211 IC50 = 429 nM T80896 D0O5KR 10060956 IC50 = 8 nM T80896 D0O6FX 10061675 IC50 = 9 nM T80896 D0P4SR 11716633 Ki = 1.3 nM T80896 D0P6FN 10125342 IC50 = 27 nM T80896 D0P7PK 77020 IC50 = 171 nM T80896 D0P8PK 10192730 IC50 = 30 nM T80896 D0R7AG 135486039 IC50 = 25 nM T80896 D0R7QY 127676 EC50 = 3700 nM T80896 D0S0SZ 135409723 IC50 = 15 nM T80896 D0S2ZJ 135430305 IC50 = 181 nM T80896 D0S6NV 10149684 IC50 = 13 nM T80896 D0S8AV 509245 IC50 = 68 nM T80896 D0S8EB 11777167 IC50 = 24 nM T80896 D0SR8Q 11458674 IC50 = 527 nM T80896 D0SY2M 5281708 Ki = 300 nM T80896 D0U0ZE 44408769 IC50 = 90 nM T80896 D0U2VA 4369550 IC50 = 5 nM T80896 D0U7KV 201385 IC50 = 11.9 nM T80896 D0UV9G 10125182 IC50 = 374 nM T80896 D0V6KJ 10214708 IC50 = 2.3 nM T80896 D0V7QZ 135528624 IC50 = 59 nM T80896 D0VN2R 10171886 IC50 = 748 nM T80896 D0W0LG 44418722 IC50 = 29 nM T80896 D0W2YR 135522274 IC50 = 963 nM T80896 D0W3FF 135503567 IC50 = 1530 nM T80896 D0W4WF 100801 IC50 = 12 nM T80896 D0W5HT 44418725 IC50 = 113 nM T80896 D0WP6A 5348729 IC50 = 1450 nM T80896 D0X0RJ 9848809 IC50 = 99 nM T80896 D0X2VK 9945207 IC50 = 2.1 nM T80896 D0X4VN 10236221 IC50 = 5 nM T80896 D0X6LK 10823890 IC50 > 5000 nM T80896 D0X7DJ 10308206 IC50 = 2.8 nM T80896 D0X7SR 10246505 EC50 = 3.5 nM T80896 D0XF9F 135484659 Ki = 1800 nM T80896 D0Y2LJ 44418729 IC50 = 37 nM T80896 D0Y4NJ 11784736 IC50 = 33.92 nM T80896 D0Y9BO 135461982 IC50 = 106 nM T80896 D0YH4T 10062042 IC50 = 3 nM T80896 D0YW4C 135494488 IC50 = 3.5 nM T80896 D0Z0UC 11638264 Ki = 1.3 nM T80896 D0ZT4U 10214633 IC50 = 7 nM T19160 D09JUG 60490 IC50 > 1000000 nM T19160 D0RA5Q 72172 IC50 > 100000 nM T19160 D00XQO 6437368 IC50 = 3900 nM T19160 D07OGR 9853400 IC50 = 1000 nM T19160 C0ZI3S 1372 IC50 = 13600 nM T19160 C71DCL 3710 IC50 = 69000 nM T19160 CS4GJ5 3711 IC50 = 57 nM T19160 CM2CV8 97908 IC50 = 42100 nM T19160 C7H3WT 127885 IC50 = 21 nM T19160 CK7IR6 155815 IC50 = 7 nM T19160 C2DIK7 155922 IC50 = 35500 nM T19160 C6TQA8 192621 IC50 = 230 nM T19160 C9RFL4 244154 IC50 = 840 nM T19160 CXTE02 381598 IC50 = 69300 nM T19160 COF19Q 885270 IC50 = 8100 nM T19160 CA96FI 1609535 IC50 = 44000 nM T19160 CLNU65 2828785 IC50 = 52000 nM T19160 CJ5B9X 3044911 IC50 = 115800 nM T19160 CDY76L 3500616 IC50 > 3300 nM T19160 C1R7KZ 9800006 IC50 = 9 nM T19160 CU79BR 9801920 IC50 = 25 nM T19160 C1BS0W 9803388 IC50 = 180 nM T19160 C8Y5QC 9804663 IC50 = 6 nM T19160 C8T2FC 9821429 IC50 = 30 nM T19160 CG9I0Z 9839929 IC50 = 25000 nM T19160 C1W9NE 9842401 IC50 = 360 nM T19160 CWS9O0 9846179 IC50 = 43 nM T19160 CA6W3U 9863966 IC50 = 11 nM T19160 C23IEK 9866653 IC50 = 125 nM T19160 C3QI5S 9867345 IC50 = 40 nM T19160 C20UBZ 9888132 IC50 = 9 nM T19160 CJT60Z 9889171 IC50 = 22 nM T19160 CO91QJ 9908515 IC50 = 28 nM T19160 CZ4UP6 9911907 IC50 = 60 nM T19160 CW04DL 9931285 IC50 = 210 nM T19160 CH2D1U 9934419 IC50 = 82 nM T19160 C9UQI6 9949943 IC50 = 4400 nM T19160 CNY1E5 9951750 IC50 = 1000 nM T19160 C9BW4J 9955004 IC50 = 8 nM T19160 CUS54H 9955690 IC50 = 6 nM T19160 CFE12L 9958280 IC50 = 250 nM T19160 CIR0H1 9984809 IC50 = 520 nM T19160 C5RL2D 9992927 IC50 > 1000000 nM T19160 C3YXB6 10006397 IC50 = 40100 nM T19160 CR3YV1 10006935 IC50 = 570 nM T19160 CZLH13 10007059 IC50 = 440 nM T19160 C7W6GZ 10016808 IC50 = 3700 nM T19160 CRS62G 10018456 IC50 > 1000000 nM T19160 CP02CV 10024065 IC50 = 900 nM T19160 C4GKM0 10048183 IC50 = 1850 nM T19160 C73GEV 10061734 IC50 > 1000000 nM T19160 C89RBI 10068833 IC50 = 430 nM T19160 CKGA81 10095448 IC50 = 3800 nM T19160 CTW2Q3 10113775 IC50 = 11 nM T19160 CNSV86 10114687 IC50 = 100 nM T19160 C1K6PG 10137047 IC50 = 11 nM T19160 CXO17P 10137777 IC50 = 108 nM T19160 C76HSK 10138016 IC50 = 806 nM T19160 CK0Y1E 10157472 IC50 = 94000 nM T19160 C6C2RG 10159102 IC50 = 10 nM T19160 C6G9WT 10160055 IC50 = 109 nM T19160 CM85ZD 10181617 IC50 = 132 nM T19160 CE3H0R 10187432 IC50 > 1600 nM T19160 C7G2VP 10202577 IC50 = 10 nM T19160 CXS1Q2 10223013 IC50 = 6 nM T19160 CB53QZ 10223158 IC50 > 1600 nM T19160 C71NJC 10223886 IC50 = 106 nM T19160 CKX5S2 10224177 IC50 = 9 nM T19160 CWG57K 10254980 IC50 = 65 nM T19160 C29IMN 10256635 IC50 = 1500 nM T19160 C46DCA 10273637 IC50 = 7 nM T19160 CB56JW 10274713 IC50 = 148 nM T19160 CE1PN2 10315432 IC50 = 390 nM T19160 CEK2Q0 10320747 IC50 = 3000 nM T19160 CX8QO3 10403265 IC50 = 5600 nM T19160 CKXQ71 10424056 IC50 > 1000000 nM T19160 C6B1NR 10432691 IC50 = 12000 nM T19160 CQZ12G 10499991 IC50 = 610 nM T19160 C4AJ0U 10503444 IC50 = 6130 nM T19160 CNF61Y 10504075 IC50 = 266 nM T19160 CZ89RL 10509638 IC50 = 2800000 nM T19160 CB2N3H 10521048 IC50 = 3000 nM T19160 C7ECZ3 10521290 IC50 = 1380 nM T19160 C8K7BR 10522189 IC50 = 620 nM T19160 CI3Y0V 10523768 IC50 = 5830 nM T19160 C2EKY3 10528351 IC50 = 4 nM T19160 CGLS04 10541824 IC50 = 8280 nM T19160 CYK50N 10542836 IC50 = 342 nM T19160 CLR3Q9 10544294 IC50 = 5880 nM T19160 CFT58W 10544972 IC50 = 321 nM T19160 C2FSP8 10546003 IC50 = 2120 nM T19160 C8C9SR 10547377 IC50 = 9430 nM T19160 C2SZ9T 10548221 IC50 = 4200 nM T19160 CEU5Q0 10548512 IC50 = 9390 nM T19160 CHS9N1 10548513 IC50 = 640 nM T19160 C2MNQ1 10548673 IC50 = 6930 nM T19160 C9BR5Z 10550162 IC50 = 1270 nM T19160 CEP53K 10550471 IC50 = 147 nM T19160 CEB1F4 10558196 IC50 = 69000 nM T19160 CD1N6Y 10564705 IC50 = 3680 nM T19160 C4YR3O 10565732 IC50 = 3610 nM T19160 C9ZTM5 10566753 IC50 = 1180 nM T19160 CUR0M3 10567842 IC50 = 7210 nM T19160 CL46SP 10567863 IC50 = 28100 nM T19160 CL38OH 10568884 IC50 = 11130 nM T19160 C0HAS8 10568956 IC50 = 420 nM T19160 C0G6KL 10569958 IC50 = 70500 nM T19160 CTF8X1 10571038 IC50 = 15220 nM T19160 C9RX7A 10571299 IC50 = 1020 nM T19160 C8PIZ5 10573509 IC50 = 450 nM T19160 CVXL13 10573634 IC50 = 23 nM T19160 CZAT67 10589888 IC50 = 1020 nM T19160 C0IE2A 10591942 IC50 = 141800 nM T19160 C2EL3Z 10592842 IC50 = 336 nM T19160 CS2H9V 10592959 IC50 = 2560 nM T19160 CHU7W3 10594135 IC50 = 96 nM T19160 C62ATP 10594151 IC50 = 52 nM T19160 CHS7U2 10594532 IC50 = 9280 nM T19160 CNB18X 10595001 IC50 = 3370 nM T19160 CG7VX1 10595053 IC50 = 180 nM T19160 CJ4S6N 10596328 IC50 = 16800 nM T19160 C32EUA 10597150 IC50 = 39 nM T19160 C8JTC0 10597699 IC50 = 51 nM T19160 CFAQ72 10598732 IC50 = 50 nM T19160 CGZ5I8 10600753 IC50 = 20 nM T19160 CDT2E5 10613668 IC50 = 2360 nM T19160 CLS0Y1 10615829 IC50 = 260 nM T19160 CHJ60E 10615830 IC50 = 34000 nM T19160 CQ0ZG6 10615906 IC50 = 550 nM T19160 CR9TL7 10618346 IC50 = 230 nM T19160 CDF5L6 10619750 IC50 = 62000 nM T19160 C3PLX0 10620311 IC50 = 8 nM T19160 C72HEB 10620653 IC50 = 1150 nM T19160 C4MF3X 10621578 IC50 = 93 nM T19160 CAX40C 10621679 IC50 = 2350 nM T19160 CWDS49 10623063 IC50 = 555 nM T19160 CUZ9B0 10623151 IC50 = 40 nM T19160 C8PX5A 10623200 IC50 = 73 nM T19160 C67CBU 10624585 IC50 = 2200 nM T19160 CF1K5S 10636392 IC50 = 38200 nM T19160 C6K5TL 10641658 IC50 = 37800 nM T19160 C30DXF 10642107 IC50 = 1360 nM T19160 CUFX41 10642850 IC50 = 860 nM T19160 C6JRI4 10644619 IC50 = 940 nM T19160 CODB20 10644711 IC50 = 77 nM T19160 CFT47L 10644791 IC50 = 203 nM T19160 CG32ZD 10645914 IC50 = 306 nM T19160 CT8HR1 10646307 IC50 = 683 nM T19160 C1BVT6 10663502 IC50 = 118 nM T19160 CUS71C 10663902 IC50 = 379 nM T19160 CC5G4O 10666583 IC50 = 527 nM T19160 CJKH86 10668302 IC50 = 85 nM T19160 C3KQP0 10687376 IC50 = 860 nM T19160 CV9T5X 10688272 IC50 = 38100 nM T19160 CCA6F5 10689154 IC50 = 390 nM T19160 CXYU62 10691131 IC50 = 1830 nM T19160 C2WH3U 10692014 IC50 = 141 nM T19160 CHR59V 10693020 IC50 = 162 nM T19160 CJWM54 10694479 IC50 = 74 nM T19160 CINZ15 10710393 IC50 = 2050 nM T19160 C28ZXB 10711124 IC50 = 74100 nM T19160 CS69EG 10712051 IC50 = 4320 nM T19160 CHGS53 10712971 IC50 = 1790 nM T19160 CCGK03 10714792 IC50 = 136 nM T19160 COSK87 10715640 IC50 = 75 nM T19160 CJ56HE 10715641 IC50 = 1270 nM T19160 C8T6KH 10716370 IC50 = 120 nM T19160 CX76RD 10717419 IC50 = 1900 nM T19160 CX0H5U 10719659 IC50 = 26 nM T19160 C6S8OH 10723410 IC50 = 75000000 nM T19160 CCEP96 10732494 IC50 = 1610 nM T19160 CGM25C 10732550 IC50 = 3700 nM T19160 CW9C1A 10735090 IC50 = 250 nM T19160 C31CAP 10735747 IC50 = 53000 nM T19160 CO84YU 10735748 IC50 = 40000 nM T19160 CER3X2 10737625 IC50 = 24 nM T19160 CTF1M8 10738557 IC50 = 121 nM T19160 C56TUC 10740804 IC50 = 1620 nM T19160 C7F4BH 10743057 IC50 = 40 nM T19160 CTSW49 10757270 IC50 = 21360 nM T19160 C07WNY 10759068 IC50 = 84700 nM T19160 C0MZ3A 10760156 IC50 = 143 nM T19160 CXN7U2 10761402 IC50 = 1380 nM T19160 C98MXS 10762842 IC50 = 5550 nM T19160 CSY8W3 10763184 IC50 = 39 nM T19160 CS95VM 10763200 IC50 = 7960 nM T19160 CFV03L 10763924 IC50 = 101200 nM T19160 CX8LW6 10764272 IC50 > 110000 nM T19160 CC19ED 10764701 IC50 = 2070 nM T19160 CB62IM 10766074 IC50 = 33 nM T19160 C3M5LB 10766584 IC50 = 16 nM T19160 CWH4X3 10782083 IC50 = 1230 nM T19160 C5D1VZ 10782159 IC50 = 1510 nM T19160 C6N1GO 10784865 IC50 = 46000 nM T19160 CEO1Y4 10784983 IC50 = 145 nM T19160 C8OBZ1 10785116 IC50 = 422 nM T19160 CXJ63K 10786018 IC50 = 6 nM T19160 C82WYB 10786028 IC50 = 12210 nM T19160 CJ0L7E 10786797 IC50 = 170 nM T19160 CR43AO 10786923 IC50 = 145 nM T19160 CB9AY2 10786935 IC50 = 59 nM T19160 CE0OY6 10787196 IC50 = 9 nM T19160 CQAG40 10787607 IC50 = 25 nM T19160 CJX69P 10788473 IC50 = 22 nM T19160 C4L3WM 10788715 IC50 = 610 nM T19160 CN0R9D 10788995 IC50 > 100000 nM T19160 C18QFO 10805784 IC50 = 1770 nM T19160 CZ2SF1 10807860 IC50 = 16700 nM T19160 CEH68P 10809342 IC50 = 230 nM T19160 CSQR04 10809782 IC50 = 15 nM T19160 C15LZY 10809862 IC50 = 25900 nM T19160 C34CGX 10810696 IC50 = 1020 nM T19160 CH7J6E 10810958 IC50 = 40200 nM T19160 CHO29M 10811318 IC50 = 44 nM T19160 C0O4XQ 10811836 IC50 = 195 nM T19160 COJR60 10814218 IC50 = 243 nM T19160 CR4O2W 10815003 IC50 = 7600 nM T19160 CLV38P 10828626 IC50 = 1230 nM T19160 C1QZY8 10829826 IC50 = 120900 nM T19160 CD2LY4 10829831 IC50 = 27180 nM T19160 CQS1A2 10830680 IC50 = 550 nM T19160 C4CK5D 10831033 IC50 = 450 nM T19160 CVQB24 10831774 IC50 = 24200 nM T19160 CPU2X6 10832199 IC50 = 1710 nM T19160 CX1Y6L 10832604 IC50 = 155 nM T19160 CW85XC 10832667 IC50 = 154 nM T19160 CH3MX7 10833045 IC50 = 46000 nM T19160 CG7V6L 10833571 IC50 = 124 nM T19160 CZ06GR 10834763 IC50 = 260 nM T19160 C9O7KE 10842569 IC50 = 4800000 nM T19160 CW0F3K 10843834 IC50 = 260000 nM T19160 C85MWA 10852262 IC50 = 64700 nM T19160 CNYX15 10852391 IC50 = 4900 nM T19160 C4UVW8 10853288 IC50 = 1180 nM T19160 C0KUR4 10853427 IC50 = 20060 nM T19160 CR09CW 10854440 IC50 = 32640 nM T19160 C60HTC 10854441 IC50 = 5320 nM T19160 C06FPE 10854831 IC50 = 910 nM T19160 CHG89F 10865991 IC50 = 12000000 nM T19160 C7LPQ2 11166515 IC50 = 73 nM T19160 CF51IR 11281695 IC50 = 82 nM T19160 CR52SA 11365008 IC50 = 7 nM T19160 C56AIM 11610604 IC50 = 300 nM T19160 C8UO0H 11734069 IC50 = 3300 nM T19160 CG1Z3I 11792248 IC50 = 360 nM T19160 CF54AN 11792751 IC50 = 9470 nM T19160 CKN4V7 11796442 IC50 > 100000 nM T19160 CXK2Q0 14530277 IC50 = 2000 nM T19160 C6RM2V 14993928 IC50 > 1660 nM T19160 C8T0ER 16135012 IC50 = 76000 nM T19160 CS59WD 16138504 IC50 = 130000 nM T19160 CPS02Y 16143405 IC50 = 100000 nM T19160 CW09CU 16144090 IC50 = 190000 nM T19160 CS8LO6 16144962 IC50 = 2400000 nM T19160 CE89KY 16157140 IC50 = 240000 nM T19160 C4F7TS 20644949 IC50 = 30 nM T19160 CI14ZM 21637538 IC50 = 15 nM T19160 C0N5TY 21920336 IC50 = 24000 nM T19160 C91UBS 24860461 IC50 = 120 nM T19160 CF5OG0 24860462 IC50 = 48 nM T19160 C4Q0JM 24860463 IC50 = 60 nM T19160 C4VM9Y 24860464 IC50 = 24 nM T19160 CD3C8T 24860465 IC50 = 39 nM T19160 CGIT86 24860466 IC50 = 52 nM T19160 C6DFQ1 24860467 IC50 = 58 nM T19160 CEV13G 24860468 IC50 = 49 nM T19160 C9HF6D 24860469 IC50 = 76 nM T19160 CZUV03 24860470 IC50 = 86 nM T19160 CR9T8M 24950865 IC50 = 100 nM T19160 CW14ZE 24950866 IC50 > 1600 nM T19160 CJD2K3 24950867 IC50 > 1600 nM T19160 CLTX47 24951184 IC50 = 14 nM T19160 C7HON4 24951342 IC50 = 35 nM T19160 CVPX65 25110662 IC50 > 1600 nM T19160 CWFM09 44298799 IC50 = 50000 nM T19160 CPY12E 44298800 IC50 = 4800 nM T19160 CHN4A0 44319936 IC50 = 2800 nM T19160 C3UF9V 44319937 IC50 = 3600 nM T19160 CWDJ03 44319952 IC50 = 2900 nM T19160 CKTG65 44320009 IC50 = 2300 nM T19160 C0HJ4E 44320172 IC50 = 5400 nM T19160 CGF1J5 44320197 IC50 = 3000 nM T19160 CPTG14 44320213 IC50 = 5200 nM T19160 CTM4D5 44320215 IC50 = 2900 nM T19160 CP1H6T 44320216 IC50 = 2100 nM T19160 CJ4X3L 44320232 IC50 = 4900 nM T19160 CZ8R2C 44320250 IC50 = 640 nM T19160 CN3Q6D 44320253 IC50 = 1800 nM T19160 CHA34O 44320336 IC50 = 240 nM T19160 CAG7P1 44322437 IC50 = 2300 nM T19160 C1GCZ3 44322473 IC50 = 3100 nM T19160 C9HGV3 44322496 IC50 = 5000 nM T19160 C2Q4YW 44322497 IC50 = 3400 nM T19160 CF6EK5 44322566 IC50 = 1700 nM T19160 CHEI15 44322593 IC50 = 350000 nM T19160 CHPU37 44323712 IC50 = 40000 nM T19160 CE1W6P 44343949 IC50 = 5300 nM T19160 CHD2O0 44343951 IC50 = 31300 nM T19160 C7SB4W 44343952 IC50 = 45800 nM T19160 CM5XT6 44344175 IC50 = 19800 nM T19160 CNL3I7 44344293 IC50 = 52900 nM T19160 C2HN4P 44365008 IC50 = 654 nM T19160 C5CAF8 44365023 IC50 = 165 nM T19160 C15UEQ 44365037 IC50 = 3680 nM T19160 CPC91X 44365039 IC50 = 58 nM T19160 CM9D8N 44365176 IC50 = 612 nM T19160 CQ53EV 44365186 IC50 = 20 nM T19160 C39YXO 44365261 IC50 = 10 nM T19160 CM28HN 44365262 IC50 = 44 nM T19160 C95JEB 44365348 IC50 = 619 nM T19160 C5UV1R 44365369 IC50 = 462 nM T19160 C4TNB9 44365370 IC50 = 15 nM T19160 CC6JR3 44365405 IC50 = 8 nM T19160 CMK04J 44365406 IC50 = 1600 nM T19160 CYX80I 44365469 IC50 = 551 nM T19160 CO3KT8 44365562 IC50 = 28 nM T19160 C9MF3W 44365563 IC50 = 49 nM T19160 CPY91D 44365634 IC50 = 33 nM T19160 CP09UQ 44365656 IC50 = 2450 nM T19160 CWA42C 44365795 IC50 = 2200000 nM T19160 CLBM81 44365796 IC50 = 4100000 nM T19160 CFRO56 44365927 IC50 = 940000 nM T19160 C7R5LV 44365928 IC50 = 5800000 nM T19160 CY79AC 44365929 IC50 = 230000 nM T19160 CH7F6Q 44410407 IC50 = 15500 nM T19160 CH1OX6 44563649 IC50 = 43700 nM T19160 CLD4I9 44578597 IC50 > 1600 nM T19160 C5SDT9 44588764 IC50 = 690 nM T19160 C4I2DU 44588787 IC50 > 1600 nM T19160 CCKD89 44588788 IC50 > 1600 nM T19160 C2L4DR 44588789 IC50 > 1600 nM T19160 C35PSA 44588790 IC50 > 1600 nM T19160 C57FJQ 44588820 IC50 > 1600 nM T19160 C0BOW3 44588821 IC50 > 1600 nM T19160 C3YWK7 51346870 IC50 = 300 nM T19160 CV19BW 53248913 IC50 = 1500 nM T19160 C5TOZ9 53248914 IC50 = 1800 nM T19160 C5RH1Q 53248940 IC50 = 2300 nM T19160 C7YJB4 53318776 IC50 = 1750 nM T19160 C32BMT 53319614 IC50 = 4200 nM T19160 CGW01A 53322243 IC50 > 1660 nM T19160 CFU46Q 53323583 IC50 = 5600 nM T19160 CSAU95 53323584 IC50 = 11670 nM T19160 C7UQC2 56658251 IC50 = 15000 nM T19160 CGHL90 56661750 IC50 = 34000 nM T19160 CN93CK 56665183 IC50 = 2800 nM T19160 CZAV62 56665184 IC50 = 6000 nM T19160 C2GR0U 56668638 IC50 = 12000 nM T19160 CK35AU 56668639 IC50 = 27000 nM T19160 CL87UJ 56668640 IC50 = 57000 nM T19160 C7LE6H 56672123 IC50 = 16000 nM T19160 C17YAM 56678854 IC50 = 2900 nM T19160 CQIV90 59871873 IC50 = 15300 nM T19160 CO4YV1 71533476 IC50 = 71000 nM T19160 CL8T6O 71568931 IC50 = 27000 nM T19160 CP5AU8 71568933 IC50 = 11500 nM T19160 CVE35U 71568934 IC50 = 5300 nM T19160 CGIA28 71569090 IC50 = 8600 nM T19160 C8HL5R 71716159 IC50 = 71000 nM T19160 CB92HR 71716414 IC50 = 217000 nM T19160 CH5WJ9 71716778 IC50 = 9200 nM T19160 C9IHB6 71717381 IC50 = 38000 nM T19160 CX48SM 71717980 IC50 = 25000 nM T19160 CW38AV 71718250 IC50 = 155000 nM T19160 C53WBM 71718251 IC50 = 85000 nM T19160 CERN41 71718857 IC50 = 262000 nM T19160 CUD01L 71719202 IC50 = 53000 nM T19160 CKM24F 71719460 IC50 = 241000 nM T19160 CT74WK 71720417 IC50 = 58000 nM T19160 C6A4SM 71720697 IC50 = 20000 nM T19160 C2EGY0 76331562 IC50 = 1800000 nM T19160 CHD26A 121596332 IC50 = 12 nM T19160 CF32QE 122197354 IC50 = 140000 nM T19160 C1VB6C 122197355 IC50 = 840000 nM T19160 C2PU7S 122197356 IC50 = 3000000 nM T19160 CPRS76 127025411 IC50 = 143 nM T19160 CHDN15 129909859 IC50 = 10 nM T19160 C8P5NZ 134693717 IC50 = 310 nM T19160 CGNA83 134812733 IC50 = 3900 nM T19160 CRMB83 135423043 IC50 = 4000 nM T19160 C80WMS 135540815 IC50 = 47700 nM T19160 CYQ02U 135540816 IC50 = 2100 nM T19160 CJI3M4 135540817 IC50 = 30500 nM T19160 C32JWI 135540836 IC50 = 8300 nM T19160 C6C2FI 135540837 IC50 = 14800 nM T19160 CJ72MG 135540865 IC50 = 29800 nM T19160 C5FZ1G 135540866 IC50 = 280 nM T19160 CHZP29 135540867 IC50 = 290 nM T19160 CT3Y7N 135540868 IC50 = 330 nM T19160 CUL9R8 135540870 IC50 = 5000 nM T19160 CB23NW 135540871 IC50 = 2200 nM T19160 C87YXS 135540872 IC50 = 76700 nM T19160 CJ2HA3 135540873 IC50 = 50900 nM T19160 CH38PY 135540874 IC50 = 11600 nM T19160 CK10WT 135540875 IC50 = 2700 nM T19160 C7H9GY 135540876 IC50 = 56000 nM T19160 C7H1AG 135540879 IC50 = 21000 nM T19160 C7VEI1 135540880 IC50 = 3100 nM T19160 CABE48 135589918 IC50 = 900 nM T19160 C7H4DL 135899007 IC50 > 100000 nM T19160 CF18ZD 135899008 IC50 > 100000 nM T19160 CZP9A0 135899009 IC50 = 5080 nM T19160 C81ZSE 135899010 IC50 > 10000 nM T19160 C5VOH2 135899011 IC50 = 10000 nM T19160 CSV1W6 135899012 IC50 = 2200 nM T19160 C7QYT2 135899013 IC50 > 100000 nM T19160 C5OV6Q 135899014 IC50 > 100000 nM T19160 C0Y9XW 135899015 IC50 = 1100 nM T19160 CE16ON 135899016 IC50 = 9000 nM T19160 CB65DI 135899017 IC50 = 4000 nM T19160 CF5DB4 135899018 IC50 = 800 nM T19160 C36RNE 135899019 IC50 = 100 nM T19160 C8IAO4 135899020 IC50 = 100 nM T19160 CUD48R 135899021 IC50 = 4500 nM T19160 CN46LC 135899022 IC50 = 3500 nM T19160 CT8Q5Z 135899023 IC50 = 2710 nM T19160 CDU7R9 135899024 IC50 = 18700 nM T19160 CB6X5L 135899025 IC50 = 5300 nM T19160 CT4GZ1 135936883 IC50 = 30 nM T19160 CQO58C 135993329 IC50 = 7600 nM T19160 C9LI3K 135993330 IC50 = 150 nM T19160 C5M8GQ 136086767 IC50 = 10000 nM T19160 CSP74T 136086768 IC50 = 970 nM T19160 C0K6PC 136086769 IC50 > 25000 nM T19160 C5ID4A 136086770 IC50 = 26000 nM T19160 C1L9PB 136086771 IC50 > 75000 nM T19160 CNG4V3 136086772 IC50 = 1300 nM T19160 C2FPV4 136086773 IC50 = 57000 nM T19160 C2H4MI 136086774 IC50 = 40700 nM T19160 C0P5CQ 136086787 IC50 = 1600 nM T19160 C5XT1S 136086788 IC50 = 2700 nM T19160 CXR85O 136086789 IC50 = 150 nM T19160 C8BDZ3 136086790 IC50 = 2700 nM T19160 CO09JG 136086791 IC50 = 330 nM T19160 CW7FC4 136086792 IC50 = 4880 nM T19160 CYAW20 136086793 IC50 > 10000 nM T19160 C4DV2Y 136086794 IC50 = 70 nM T19160 C4A6JO 136086795 IC50 = 220 nM T19160 C7AH6F 136086796 IC50 = 3250 nM T19160 C4TMB9 136086797 IC50 = 50 nM T19160 C83KHP 136086798 IC50 = 2040 nM T19160 CH7JU1 136086799 IC50 = 290 nM T19160 CS0XK3 136086800 IC50 = 3040 nM T19160 CB2O1N 136086801 IC50 = 580 nM T19160 C2VU8G 136086802 IC50 = 230 nM T19160 CN2K0P 136086803 IC50 = 30000 nM T19160 C4PE6L 136086804 IC50 = 1700 nM T19160 C02CUW 137704643 IC50 = 38 nM T19160 CHG3A9 141721984 IC50 = 11 nM T19160 COK2V0 141721987 IC50 = 70 nM T19160 C9G0YT 141721988 IC50 = 110 nM T19160 CQW3U8 141721990 IC50 = 190 nM T19160 CHQ8T0 141721991 IC50 = 910 nM T19160 CY0CD2 141721992 IC50 = 21 nM T19160 CIJ89F 145950092 IC50 = 5700 nM T19160 CMF6V0 145951004 IC50 = 2300 nM T19160 CZ0GL9 145952337 IC50 = 3900 nM T19160 C39QIE 145958640 IC50 = 3600 nM T19160 CPR0E9 145966028 IC50 = 290 nM T19160 C36PXF 145966065 IC50 = 57 nM T19160 C5UJ2P 145966281 IC50 = 4000 nM T19160 C2HSB3 145966662 IC50 = 820 nM T19160 CK9FV5 145972205 IC50 = 890 nM T19160 C9L2IH 145972643 IC50 > 10000 nM T19160 C4EZY7 145973101 IC50 = 470 nM T19160 C8RFM3 145973261 IC50 = 630 nM T19160 C39GPD 145974999 IC50 = 4400 nM T19160 C1L4CT 145975332 IC50 = 4500 nM T19160 CMB21Z 145975404 IC50 = 1200 nM T19160 CS8A5G 145975567 IC50 = 140 nM T19160 CLM80S 145975768 IC50 = 170 nM T19160 C95DNK 145975863 IC50 = 92 nM T19160 CD90YF 145975932 IC50 = 1900 nM T19160 C20XUS 145978713 IC50 = 3100 nM T19160 CU4ME9 145978748 IC50 = 44 nM T19160 C28ITA 155523326 IC50 = 18 nM T19160 D02AYI 11031651 IC50 = 7300 nM T19160 D02GTZ 44410505 IC50 = 23200 nM T19160 D02IVU 21774960 IC50 = 3000 nM T19160 D03BAB 23243376 IC50 = 1400 nM T19160 D05LWK 44410408 IC50 = 63900 nM T19160 D07VJT 23661736 IC50 = 19900 nM T19160 D0B9VV 10386285 IC50 = 4300 nM T19160 D0C8MT 260806 IC50 = 52500 nM T19160 D0J2EE 9957245 IC50 = 1600 nM T19160 D0L6GV 11962186 IC50 = 3000 nM T19160 D0O2DQ 237 IC50 = 76000000 nM T19160 D0P1LP 7090 IC50 > 1000000 nM T10918 CUZC83 5308428 EC50 = 497 nM T10918 CY7O0L 53378752 IC50 = 226 nM T10918 CS13DM 121277209 EC50 = 213 nM T10918 C9C5BR 121277212 EC50 = 314 nM T10918 CV83UW 121279842 EC50 = 90 nM T17569 D03DAP 3356 IC50 = 51000 nM T17569 D04OSE 4485 IC50 = 6100 nM T17569 D0X4RN 3676 IC50 = 2188000 nM T17569 D00BUR 216327 IC50 > 1000 nM T17569 D02AIN 122678117 IC50 > 32000 nM T17569 D04LOR 51030730 IC50 = 46 nM T17569 D0K9IF 71666749 IC50 > 30000 nM T17569 D0S5IR 86294073 IC50 > 30000 nM T17569 D0OS6O 60149 IC50 = 2000 nM T17569 CI7BE6 219025 IC50 = 2370 nM T17569 CLD6J9 441074 IC50 = 7300 nM T17569 CZN6S9 743974 IC50 > 50118.72 nM T17569 CW1TI4 2728088 IC50 = 4720 nM T17569 CY78UB 2728090 IC50 = 5450 nM T17569 CDUR91 2728127 IC50 = 8370 nM T17569 C57QVA 2747476 IC50 = 38780 nM T17569 CGS07D 2747486 IC50 = 37500 nM T17569 CNXW51 4224660 IC50 = 3200 nM T17569 C9INQ8 4390854 IC50 > 30000 nM T17569 CWU84K 4998225 IC50 = 109740 nM T17569 C6HA8E 5388709 IC50 > 30000 nM T17569 C8W2QA 6439099 IC50 = 7600 nM T17569 CO9NP6 6890860 IC50 = 810 nM T17569 CSA4X5 9259741 IC50 = 16110 nM T17569 C07NPJ 9259759 IC50 = 10130 nM T17569 C4M2HZ 9259800 IC50 = 28570 nM T17569 C5C4UF 9260142 IC50 = 5020 nM T17569 C5Y8AR 9260156 IC50 = 2620 nM T17569 C3I0KG 9260177 IC50 = 4380 nM T17569 CDN9G6 9434363 IC50 = 29420 nM T17569 CML41X 9434371 IC50 = 3590 nM T17569 CT3W6H 9801960 IC50 = 4500 nM T17569 C9JWG5 9825229 IC50 = 2800 nM T17569 C7UGB8 9826037 IC50 = 700 nM T17569 CGBE91 9827303 IC50 = 1200 nM T17569 CL34VA 9827609 IC50 = 260 nM T17569 CPQL48 9827686 IC50 > 10000 nM T17569 C30IAQ 9840150 IC50 = 190 nM T17569 CN0UB8 9841529 IC50 = 7100 nM T17569 CG1DH8 9847973 IC50 = 160 nM T17569 C3Y6DL 9848021 IC50 = 260 nM T17569 CQ7J5I 9870026 IC50 = 1200 nM T17569 CO42SU 9889729 IC50 = 600 nM T17569 COKF63 9906009 IC50 = 200 nM T17569 CGKT80 9908970 IC50 = 4100 nM T17569 CA53RP 9910831 IC50 = 5600 nM T17569 C0JNF1 9915801 IC50 = 316 nM T17569 C4CH5D 9927877 IC50 = 1300 nM T17569 C29ZMV 9931732 IC50 = 3300 nM T17569 C40KYF 9932430 IC50 = 800 nM T17569 CC3H8U 9954715 IC50 = 2600 nM T17569 C1N5LX 10065677 IC50 = 7700 nM T17569 C97OQC 10088458 IC50 = 4300 nM T17569 C0UY8K 10159855 IC50 = 2600 nM T17569 CT19IQ 10162503 IC50 = 700 nM T17569 CTIV71 10228115 IC50 = 8500 nM T17569 C2OK7Y 10272874 IC50 = 5000 nM T17569 CUFL28 10274235 IC50 = 400 nM T17569 CZN82G 10406083 IC50 = 3600 nM T17569 CVL5Y3 10875427 IC50 = 9100 nM T17569 CZFJ03 10899797 IC50 > 60000 nM T17569 CYC4S6 10928160 IC50 = 7000 nM T17569 CGUA38 10939752 IC50 = 2400 nM T17569 CCR96E 10940235 IC50 = 11200 nM T17569 C20UNS 11038129 IC50 = 1000 nM T17569 CDJ13N 11059094 IC50 = 7800 nM T17569 C07NWJ 11059860 IC50 = 300 nM T17569 C0V5IR 11070755 IC50 = 300 nM T17569 CZ1W0R 11101439 IC50 = 4000 nM T17569 C25HLY 11114384 IC50 = 7700 nM T17569 CZ81UG 11123576 IC50 = 2200 nM T17569 CAM6Y1 11146287 IC50 = 4800 nM T17569 CDY8S7 11165745 IC50 = 790 nM T17569 CDOC09 11199458 IC50 = 870 nM T17569 C9X0TH 11291017 IC50 = 680 nM T17569 C0PUK5 11360073 IC50 = 160 nM T17569 CWO2A7 11382160 IC50 = 690 nM T17569 CU7B8I 11525190 IC50 = 9 nM T17569 C8NM2I 11538313 EC50 = 5000 nM T17569 C12VCK 11573765 IC50 = 284 nM T17569 C47TZG 11595633 IC50 = 206 nM T17569 CAU61Q 11610483 IC50 = 517 nM T17569 CA5W9R 11618060 EC50 = 900 nM T17569 CCE90V 11638319 IC50 = 850 nM T17569 CEXK54 11653686 IC50 = 4946 nM T17569 CR92TH 11660563 IC50 = 583 nM T17569 C9K3EO 11688027 IC50 > 60000 nM T17569 CFGR63 11695646 IC50 = 2222 nM T17569 CLT3Z7 11695929 EC50 = 700 nM T17569 CZ9SY1 11702625 IC50 = 2140 nM T17569 C2L1CA 11732025 IC50 = 3500 nM T17569 C90VTJ 11826160 IC50 = 12000 nM T17569 CU6E3R 11826630 IC50 = 1000 nM T17569 CNCV28 11827109 IC50 = 1700 nM T17569 C0SMQ3 11995420 IC50 = 1010 nM T17569 C9KSG8 11995421 IC50 = 250 nM T17569 CEYB03 11995422 IC50 = 60 nM T17569 C58BPD 11995424 IC50 = 260 nM T17569 CTYE90 11995521 IC50 = 120 nM T17569 C0DE5H 11995522 IC50 = 1050 nM T17569 CE9AT3 12653729 IC50 = 252 nM T17569 CD34SB 15982534 IC50 > 100000 nM T17569 C3JT4R 16007209 IC50 = 294 nM T17569 CB64EN 16049818 IC50 = 21 nM T17569 CSEA12 16049867 IC50 = 150 nM T17569 CO2S6X 16050462 IC50 = 43 nM T17569 CLR07F 16050659 IC50 = 219 nM T17569 C13PZH 16050755 IC50 = 187 nM T17569 CPZ80C 16050947 IC50 = 198 nM T17569 C8C1FL 16050950 IC50 = 24 nM T17569 CO5VF2 16050952 IC50 = 22 nM T17569 CYNL61 16050953 IC50 = 118 nM T17569 CU3JF5 16051050 IC50 = 73 nM T17569 C6NLQ9 16051053 IC50 = 197 nM T17569 CL48DJ 16067577 IC50 = 184 nM T17569 CGP0J6 16067578 IC50 = 137 nM T17569 CK94WY 16067666 IC50 = 266 nM T17569 C15YUI 16067667 IC50 = 3836 nM T17569 CGV37P 16067668 IC50 = 708 nM T17569 COK93T 16067762 IC50 = 6348 nM T17569 C4X9WF 16067864 IC50 = 250 nM T17569 CAD3H8 16067970 IC50 = 490 nM T17569 CLUV52 16067971 IC50 = 100 nM T17569 CZ52CY 16067972 IC50 = 36 nM T17569 CECT12 16067973 IC50 = 94 nM T17569 C2P1GF 16067974 IC50 = 252 nM T17569 CCU3P1 16067975 IC50 = 362 nM T17569 C25JRI 16068075 IC50 = 353 nM T17569 CFJ8R5 16068078 IC50 = 341 nM T17569 CE7CP4 16068080 IC50 = 240 nM T17569 CT8W3J 16068194 IC50 = 498 nM T17569 C4JCO2 16068195 IC50 = 256 nM T17569 CX3G4D 16068198 IC50 = 757 nM T17569 CZ5QK7 16068305 IC50 = 298 nM T17569 CV4WU7 16068309 IC50 = 283 nM T17569 CYEH75 16068516 IC50 = 432 nM T17569 CB1XC9 16068517 IC50 = 589 nM T17569 C9OJ0P 16068518 IC50 = 249 nM T17569 CR98NG 16068621 IC50 = 1594 nM T17569 C72XJF 16068622 IC50 = 410 nM T17569 C9S7IC 16068624 IC50 = 3379 nM T17569 C7VQ2G 16068728 IC50 = 326 nM T17569 CU7Q5L 16068729 IC50 = 147 nM T17569 CGJQ19 16068833 IC50 = 2669 nM T17569 CESK71 16068836 IC50 = 6868 nM T17569 C2DRM7 16068839 IC50 = 5323 nM T17569 CZ4H7M 16068947 IC50 = 13760 nM T17569 CH8WZ9 16102139 IC50 = 23 nM T17569 CYF7U1 16662313 IC50 = 90 nM T17569 C6OBK5 16722240 IC50 = 110 nM T17569 CS14WU 16722242 IC50 = 171 nM T17569 C8T4JF 16722295 IC50 = 11 nM T17569 CDU3E0 17474273 IC50 = 4230 nM T17569 CY9QV3 17748224 IC50 = 33 nM T17569 C1GUE6 17752926 IC50 = 60 nM T17569 CYB69N 18134053 IC50 = 9130 nM T17569 CZ40KV 18134054 IC50 = 29340 nM T17569 CHFV68 18134055 IC50 = 5180 nM T17569 CO17PU 21635104 IC50 = 200 nM T17569 C02YIQ 24963478 IC50 = 1100 nM T17569 CQ58IV 24964189 IC50 = 1500 nM T17569 CS6XP4 24964190 IC50 = 900 nM T17569 C6Z7KY 24967023 IC50 = 7600 nM T17569 C14KJT 24967024 IC50 = 4500 nM T17569 CY02UG 24967383 IC50 = 2400 nM T17569 CV40UK 24967750 IC50 = 2700 nM T17569 C4X1JN 24968454 IC50 = 1200 nM T17569 CYH04T 24968455 IC50 = 1300 nM T17569 C4D2VI 24968798 IC50 = 2100 nM T17569 CV02TA 25017750 IC50 = 240 nM T17569 CTYD20 25018000 IC50 = 240 nM T17569 CJNR78 25018002 IC50 = 250 nM T17569 C9AKD7 25018252 IC50 = 160 nM T17569 CB36TF 25019018 IC50 = 330 nM T17569 CUF48R 25019019 IC50 = 610 nM T17569 C91QFN 25019282 IC50 = 480 nM T17569 CYG87R 27847327 IC50 = 5500 nM T17569 CA0W3I 28222848 IC50 = 4490 nM T17569 CI2RH1 31692234 IC50 = 9100 nM T17569 CX76VJ 44219755 IC50 = 90 nM T17569 CB04SM 44289875 IC50 ~ 2900 nM T17569 CG19SR 44327873 IC50 = 3500 nM T17569 CV1TA9 44327874 IC50 = 9000 nM T17569 CDT2M6 44327918 IC50 = 1700 nM T17569 CS17ID 44327919 IC50 = 3100 nM T17569 C5J1VM 44327920 IC50 = 10000 nM T17569 C1RO7D 44327937 IC50 = 600 nM T17569 C09QDX 44327941 IC50 = 700 nM T17569 CE52TF 44328123 IC50 = 6500 nM T17569 C4IOT7 44328125 IC50 = 6200 nM T17569 CMY67Z 44328134 IC50 = 3800 nM T17569 CXL40O 44328260 IC50 = 2700 nM T17569 CNS9J6 44328262 IC50 = 1600 nM T17569 C5WXP6 44328272 IC50 = 500 nM T17569 C5JO9M 44328281 IC50 = 2200 nM T17569 C6NAP7 44328282 IC50 = 1200 nM T17569 CWTA09 44328298 IC50 = 500 nM T17569 C28RVI 44328299 IC50 = 1900 nM T17569 CX0LS1 44328315 IC50 = 6900 nM T17569 CG94NW 44364149 IC50 = 9500 nM T17569 CN1EX7 44415895 IC50 = 137 nM T17569 CMYJ86 44418028 IC50 = 330 nM T17569 CHP7D4 44418031 IC50 = 370 nM T17569 C0Z1BI 44418048 IC50 = 400 nM T17569 C7US9W 44418049 IC50 = 180 nM T17569 COT0S9 44418057 IC50 = 1310 nM T17569 CB74SR 44418071 IC50 = 368 nM T17569 CEY65I 44418075 IC50 = 265 nM T17569 C5KB2U 44418086 IC50 = 550 nM T17569 C5ISB7 44418087 IC50 = 330 nM T17569 CGV26X 44418088 IC50 = 215 nM T17569 C91KCR 44418095 IC50 = 1773 nM T17569 C45WSY 44418096 IC50 = 113 nM T17569 C7N0BS 44418101 IC50 = 3698 nM T17569 C2GXD0 44418117 IC50 = 187 nM T17569 C9N5LU 44418118 IC50 = 113 nM T17569 CT16WE 44418119 IC50 = 95 nM T17569 CG3LM9 44418123 IC50 = 150 nM T17569 C61BYQ 44418124 IC50 = 812 nM T17569 C9N6TB 44418140 IC50 = 390 nM T17569 CL4P2S 44418142 IC50 = 380 nM T17569 CJ8UL2 44418144 IC50 = 162 nM T17569 C1ZPJ0 44418146 IC50 = 69 nM T17569 C51JFR 44418148 IC50 = 179 nM T17569 CJRO39 44418167 IC50 = 269 nM T17569 CA9IU3 44418172 IC50 = 487 nM T17569 CQMN19 44418173 IC50 = 204 nM T17569 CZO90U 44418196 IC50 = 177 nM T17569 CI04UY 44418199 IC50 = 207 nM T17569 CH95LR 44418204 IC50 = 480 nM T17569 C39ZBV 44418205 IC50 = 537 nM T17569 C0VZ5H 44418247 IC50 = 463 nM T17569 C7TC3Y 44426322 IC50 = 290 nM T17569 CB7AI0 44426323 IC50 = 281 nM T17569 C0I6CQ 44426324 IC50 = 170 nM T17569 CPT28O 44426325 IC50 = 77 nM T17569 CY0IZ1 44426326 IC50 = 130 nM T17569 C52MHS 44426327 IC50 = 170 nM T17569 CC2L5X 44426328 IC50 = 210 nM T17569 CFEP20 44426329 IC50 = 79 nM T17569 CI5JQ0 44426330 IC50 > 1000 nM T17569 C57CFR 44426332 IC50 > 10000 nM T17569 CJSA29 44426333 IC50 > 1000 nM T17569 CO3K4E 44426334 IC50 = 200 nM T17569 C1FTM2 44426336 IC50 = 400 nM T17569 C85DFL 44426340 IC50 = 340 nM T17569 CB79PX 44426342 IC50 = 150 nM T17569 C8NGE5 44426346 IC50 > 1000 nM T17569 C37PWI 44426349 IC50 > 1000 nM T17569 C1J7FC 44426353 IC50 > 1000 nM T17569 CSPC40 44426357 IC50 = 57 nM T17569 CM1QG0 44426360 IC50 = 320 nM T17569 CFN6Q5 44426361 IC50 = 120 nM T17569 C23NQI 44426362 IC50 = 130 nM T17569 CWI2B3 44426363 IC50 = 120 nM T17569 CG50QZ 44426364 IC50 = 280 nM T17569 C4E9FS 44426392 IC50 > 1000 nM T17569 CE5G0B 44426393 IC50 = 260 nM T17569 C3I0RJ 44426394 IC50 = 89 nM T17569 CB5KR0 44426395 IC50 = 200 nM T17569 CM7B1D 44426396 IC50 = 220 nM T17569 CGU51D 44426397 IC50 = 110 nM T17569 C69HXQ 44426398 IC50 = 240 nM T17569 CAP18U 44426399 IC50 > 10000 nM T17569 CF6M8H 44426400 IC50 = 510 nM T17569 C8F3ZQ 44439688 IC50 = 760 nM T17569 CLO5I0 44439690 IC50 = 880 nM T17569 CNF52R 44439694 IC50 = 150 nM T17569 C98RYZ 44439695 IC50 = 300 nM T17569 CO84EZ 44439696 IC50 = 440 nM T17569 CYB37A 44439697 IC50 = 200 nM T17569 CU34VJ 44439698 IC50 = 240 nM T17569 CU4G5P 44450515 IC50 = 912 nM T17569 CK8TN2 44450516 IC50 = 776 nM T17569 C0FW1K 44450530 IC50 = 649 nM T17569 CULO37 44450539 IC50 = 378 nM T17569 CU84IE 44450556 IC50 = 2090 nM T17569 CA0BZ3 44450557 IC50 = 1560 nM T17569 CH89QB 44450558 IC50 = 615 nM T17569 CQ62WH 44450567 IC50 = 605 nM T17569 C9LC8X 44450682 IC50 = 46 nM T17569 C6IK7J 44541892 IC50 = 7450 nM T17569 C16HIP 44542338 IC50 = 200 nM T17569 C2B6OY 44542339 IC50 = 100 nM T17569 CQ4W7V 44542340 IC50 = 560 nM T17569 CN64WQ 44544347 IC50 = 1500 nM T17569 C3OK2I 44573922 IC50 = 220 nM T17569 C7D2EB 44573924 IC50 = 290 nM T17569 C7ZFT0 44573925 IC50 = 300 nM T17569 CWDM60 44574029 IC50 = 430 nM T17569 CMNA45 44574030 IC50 = 160 nM T17569 CM8DS7 44574049 IC50 = 70 nM T17569 C70NZD 44574085 IC50 = 3000 nM T17569 CCIQ65 44574163 IC50 = 450 nM T17569 CV64TR 44574164 IC50 = 450 nM T17569 C2V8UL 44574185 IC50 = 710 nM T17569 CJH08W 44574186 IC50 = 340 nM T17569 CZE9H7 44574187 IC50 = 640 nM T17569 C3Y4GH 44574215 IC50 = 250 nM T17569 CE46UH 44574244 IC50 = 200 nM T17569 CC0W9Q 44574245 IC50 = 430 nM T17569 C1CW8S 44574246 IC50 = 350 nM T17569 C3JP2W 44574247 IC50 = 230 nM T17569 C53EPX 44574274 IC50 = 610 nM T17569 CJIL50 44574275 IC50 = 590 nM T17569 CKN3Y2 44574276 IC50 = 280 nM T17569 CMQ17N 45484111 IC50 = 520 nM T17569 C5YT2N 45484113 IC50 = 340 nM T17569 C85XBW 45484115 IC50 = 770 nM T17569 C9D6SC 45484116 IC50 = 230 nM T17569 CO42HZ 45484117 IC50 = 900 nM T17569 CJE36D 45484118 IC50 = 600 nM T17569 C9L4KT 46205341 IC50 > 333000 nM T17569 CL41FE 46206000 IC50 > 100000 nM T17569 C4ST0I 46448745 IC50 = 3970 nM T17569 C1TXI0 46885514 IC50 > 60000 nM T17569 CKF74T 46885587 IC50 = 234 nM T17569 CKH5W7 46885611 IC50 = 7935 nM T17569 C10CAI 50908735 IC50 = 540 nM T17569 CNP3Q6 50908736 IC50 = 480 nM T17569 CP3D8F 51030551 IC50 = 210 nM T17569 C0QG2E 51030636 IC50 = 90 nM T17569 C4UPJ2 51030637 IC50 = 80 nM T17569 C6GC4D 51030638 IC50 = 170 nM T17569 C7NQV1 51030641 IC50 = 250 nM T17569 CKZ23X 51030643 IC50 = 150 nM T17569 CSE2G4 51030732 IC50 = 110 nM T17569 CM1F2R 51030830 IC50 = 100 nM T17569 CWQ20B 51030833 IC50 = 100 nM T17569 CSR8Z9 51183445 IC50 = 10170 nM T17569 C7EB3O 52941155 IC50 = 830 nM T17569 CVB2S3 52941198 IC50 = 560 nM T17569 CU23TL 52941375 IC50 = 1180 nM T17569 CH29GZ 52941394 IC50 = 1350 nM T17569 CG2TW3 52941465 IC50 = 350 nM T17569 CYU9F4 52941559 IC50 = 450 nM T17569 CS1C3E 52941613 IC50 = 5970 nM T17569 CBJ50X 52942519 IC50 > 50000 nM T17569 CH7KN9 52942767 IC50 = 730 nM T17569 C84XGP 52943813 IC50 = 1320 nM T17569 CW9DO1 52943894 IC50 = 370 nM T17569 C9VHK1 52943985 IC50 = 2640 nM T17569 CB96VD 52944057 IC50 = 780 nM T17569 C5CN7Y 52944792 IC50 = 440 nM T17569 CIW8Q2 52944838 IC50 = 1390 nM T17569 CQ02KD 52944866 IC50 = 2880 nM T17569 C1PAQ4 52944957 IC50 = 410 nM T17569 CN35LH 52944958 IC50 = 360 nM T17569 C9PX5E 52944999 IC50 = 340 nM T17569 C3DYJ5 52945000 IC50 = 290 nM T17569 C0O4CT 52945029 IC50 = 520 nM T17569 C0AFU8 52945163 IC50 = 320 nM T17569 CIN90C 52946106 IC50 > 50000 nM T17569 CV31NF 52946270 IC50 = 270 nM T17569 CIV24B 52946310 IC50 = 13900 nM T17569 CX8C5G 52946322 IC50 > 50000 nM T17569 C4ED8W 52946335 IC50 = 790 nM T17569 C8R1ZO 52946384 IC50 = 370 nM T17569 CJ7AY2 52946550 IC50 = 9060 nM T17569 C9WRK4 52947357 IC50 = 13700 nM T17569 C28QEH 52948441 IC50 = 630 nM T17569 CJ1RH6 52948489 IC50 = 960 nM T17569 CU89SW 52948510 IC50 = 1980 nM T17569 CMG1Z5 52948605 IC50 = 2000 nM T17569 C0LCS3 52948698 IC50 = 490 nM T17569 CZT6C4 52948768 IC50 > 50000 nM T17569 C4IL2V 52948983 IC50 = 900 nM T17569 CAB7U5 52948996 IC50 = 320 nM T17569 CF6U3A 52949881 IC50 > 50000 nM T17569 C46JBA 52949924 IC50 = 2220 nM T17569 C43YBI 52949966 IC50 = 240 nM T17569 C1FOZ0 52949971 IC50 = 460 nM T17569 C23WVS 53361524 IC50 > 33300 nM T17569 CD8P9A 55483031 IC50 = 3390 nM T17569 CONA69 57065698 IC50 = 2250 nM T17569 C4VT6Z 58615686 IC50 = 9950 nM T17569 C2D3HQ 60168069 IC50 > 100000 nM T17569 C5BU7L 66829310 IC50 = 41 nM T17569 CPZQ50 66829372 IC50 = 579 nM T17569 C38BYQ 66829396 IC50 = 64 nM T17569 CEVJ65 66829417 IC50 = 84 nM T17569 CBE2J9 66829485 IC50 = 133 nM T17569 CQF8M5 66829565 IC50 = 1592 nM T17569 CRI63W 66829595 IC50 = 33 nM T17569 CD1BQ8 66829616 IC50 = 23 nM T17569 C8OZR1 66829709 IC50 = 30 nM T17569 CEQ7A6 66829716 IC50 = 2865 nM T17569 CMAD65 66829757 IC50 = 136 nM T17569 CJMU80 67055888 IC50 = 50 nM T17569 CC62HR 67264671 IC50 > 10000 nM T17569 CKQ9W2 67264691 IC50 = 1386 nM T17569 C3F2JN 67264841 IC50 = 1276 nM T17569 C38ROH 67264950 IC50 = 444 nM T17569 C3CAR6 67265132 IC50 = 64 nM T17569 C3K4RT 68204896 IC50 = 60 nM T17569 CWTD61 68204898 IC50 = 50 nM T17569 CF59AG 68204902 IC50 = 90 nM T17569 CLS7H4 68204905 IC50 = 120 nM T17569 CG0X2O 68204906 IC50 = 160 nM T17569 CM58CG 68204907 IC50 = 40 nM T17569 CRN5M3 68204912 IC50 = 130 nM T17569 CNTP78 68204921 IC50 = 330 nM T17569 CWT8R0 68204939 IC50 = 80 nM T17569 C7V2SY 68204942 IC50 = 100 nM T17569 CTL0O6 68770301 IC50 = 1400 nM T17569 CUVF59 68770356 IC50 = 2200 nM T17569 CT2D3M 68772321 IC50 = 700 nM T17569 CX5Q2G 68772765 IC50 = 800 nM T17569 CM92FU 68773430 IC50 = 3500 nM T17569 CZ07NC 68773726 IC50 = 37000 nM T17569 C16VTD 68774064 IC50 = 6900 nM T17569 CR28FH 68774353 IC50 = 13000 nM T17569 CWV13E 68774423 IC50 = 11300 nM T17569 C5J1XL 68774942 IC50 = 1400 nM T17569 C59FDP 68775014 IC50 = 1100 nM T17569 CTD8Q5 68775141 IC50 = 900 nM T17569 C23PDV 68775184 IC50 = 900 nM T17569 CL6N2D 68775231 IC50 = 400 nM T17569 CC98XW 68775928 IC50 = 6000 nM T17569 CR37DA 71419478 IC50 = 300 nM T17569 C5SML3 71449452 IC50 = 200 nM T17569 COQ0P1 71453071 IC50 = 600 nM T17569 CLE21W 71520368 IC50 = 11000 nM T17569 C5S0FT 71520369 IC50 = 17000 nM T17569 CZY20B 71520370 IC50 = 4100 nM T17569 C0T9BG 71520371 IC50 = 2300 nM T17569 C3AKL4 71520372 IC50 = 1600 nM T17569 C4OBM9 71520373 IC50 = 530 nM T17569 CXT3L0 71520486 IC50 = 1900 nM T17569 CA3B5V 71520487 IC50 = 1300 nM T17569 C1HI9J 71520488 IC50 = 1000 nM T17569 C92QDP 71520489 IC50 = 590 nM T17569 CM6DZ1 71520490 IC50 = 200 nM T17569 CD1XT8 71520491 IC50 = 930 nM T17569 CU23JX 71520492 IC50 = 180 nM T17569 CSQH86 71520575 IC50 = 620 nM T17569 C6TO3P 71520576 IC50 = 100 nM T17569 C0WC7P 71520577 IC50 = 140 nM T17569 CZ0QX1 71520578 IC50 = 750 nM T17569 CWAO49 71604376 IC50 = 16070 nM T17569 C8G6PW 71716112 IC50 = 540 nM T17569 COBD81 71716733 IC50 = 120 nM T17569 CY8AS2 71717330 IC50 = 80 nM T17569 C2TM0Z 71719149 IC50 = 330 nM T17569 CB0WC3 71719150 IC50 = 2700 nM T17569 CS43PH 72205298 IC50 = 38730 nM T17569 CJ7AH3 72205299 IC50 = 3930 nM T17569 C9LA4P 72205300 IC50 = 12920 nM T17569 CA5OB3 72205302 IC50 = 3560 nM T17569 CA10KU 72205492 IC50 = 1720 nM T17569 C78TDP 72205494 IC50 = 2380 nM T17569 CB19LS 72205495 IC50 = 3140 nM T17569 C3I1WO 72205678 IC50 = 6210 nM T17569 C3AI8D 72205680 IC50 = 185140 nM T17569 C1REI7 72205885 IC50 = 6450 nM T17569 C7CHK8 72205888 IC50 = 65420 nM T17569 C1LFU2 73346537 IC50 = 1900 nM T17569 CB3K2X 73346538 IC50 = 11240 nM T17569 CKH6L4 73346539 IC50 = 16910 nM T17569 C5EJ6B 73348019 IC50 = 1520 nM T17569 CX08AE 73349556 IC50 = 510 nM T17569 CC5B9P 73351121 IC50 = 740 nM T17569 CZ15AU 73351122 IC50 = 2180 nM T17569 CC20XL 73351123 IC50 = 24010 nM T17569 CTLF48 73351124 IC50 = 1770 nM T17569 CP3V8S 73352588 IC50 = 2140 nM T17569 CC3E6P 73354082 IC50 = 3730 nM T17569 C5LBH4 73357152 IC50 = 250 nM T17569 C7EXL1 76311070 IC50 = 2700 nM T17569 CNKW61 76311071 IC50 > 10000 nM T17569 CO1TF8 76311072 IC50 = 210 nM T17569 CR0J4Y 76311073 IC50 = 8800 nM T17569 CCN4Q7 76311074 IC50 > 30000 nM T17569 C3V8QA 76311075 IC50 = 8700 nM T17569 C7G0SH 76314696 IC50 = 7600 nM T17569 C4RVF2 76314697 IC50 = 8700 nM T17569 CA9Z2P 76318265 IC50 = 2000 nM T17569 C8JRZ9 76318266 IC50 > 10000 nM T17569 C29SUN 76318267 IC50 = 7200 nM T17569 CXU8E0 76321967 IC50 = 28000 nM T17569 CK13YQ 76321968 IC50 = 810 nM T17569 CY6MU9 76321969 IC50 = 2200 nM T17569 CD8PJ1 76321970 IC50 = 2000 nM T17569 C6QI2C 76321971 IC50 = 800 nM T17569 CL6H1G 76321972 IC50 > 30000 nM T17569 C3F0UK 76325592 IC50 > 10000 nM T17569 CGF1Z5 76325593 IC50 = 2600 nM T17569 CA2C8Q 76329153 IC50 = 4800 nM T17569 CK5G2T 76329154 IC50 = 4100 nM T17569 C05ZMU 76332813 IC50 = 2200 nM T17569 CP20RQ 76336433 IC50 = 2800 nM T17569 CUKY70 76336434 IC50 = 4300 nM T17569 C02YVP 76336435 IC50 = 8100 nM T17569 C2JWB6 76336436 IC50 = 2000 nM T17569 CN74YH 78788985 IC50 = 720 nM T17569 C6GS7X 78788989 IC50 = 21920 nM T17569 CWRN76 78795764 IC50 = 9740 nM T17569 C6CD1Z 86617892 IC50 = 10500 nM T17569 CH86IJ 86670613 IC50 = 70 nM T17569 CJ29DT 86977989 IC50 = 13530 nM T17569 CRT2P3 90643635 IC50 = 48360 nM T17569 C4W7JE 90643636 IC50 = 1520 nM T17569 CMFW64 90643637 IC50 = 6440 nM T17569 C1FT9B 90643638 IC50 = 25270 nM T17569 C94KHQ 90643639 IC50 = 7140 nM T17569 CG7WJ6 90643640 IC50 = 4510 nM T17569 CM9T7F 90643641 IC50 = 56750 nM T17569 CPL5Q9 90643642 IC50 = 11820 nM T17569 CS0DM4 90643643 IC50 = 7330 nM T17569 C26PLG 90643644 IC50 = 14460 nM T17569 CGDQ14 90643645 IC50 = 8930 nM T17569 CHJ1L8 90643646 IC50 = 1240 nM T17569 CXQ76K 90643647 IC50 = 17160 nM T17569 CB06NO 90643648 IC50 = 50240 nM T17569 CG8U0B 90643649 IC50 = 85930 nM T17569 CI2VA6 90643650 IC50 = 63180 nM T17569 CLJ87B 90643651 IC50 = 2290 nM T17569 CH01QZ 90643652 IC50 = 970 nM T17569 COY15C 90643653 IC50 = 68030 nM T17569 C1DTE9 90643654 IC50 = 12710 nM T17569 C4MS2G 90643655 IC50 = 12180 nM T17569 C2JAQ6 90643656 IC50 = 1480 nM T17569 C0B7LH 90645435 IC50 = 88 nM T17569 CXU7O2 90645436 IC50 = 138 nM T17569 CGA98E 90645438 IC50 = 784 nM T17569 CQSZ72 90675942 IC50 > 30000 nM T17569 CTBD74 90675943 IC50 > 30000 nM T17569 CM12LR 102597975 IC50 = 6100 nM T17569 C1YK2E 122678192 IC50 > 32000 nM T17569 C0A5RC 127031270 IC50 = 500 nM T17569 COD4E0 127031330 IC50 = 1200 nM T17569 CM89VC 127031576 IC50 > 10000 nM T17569 C98TDU 127031577 IC50 > 32000 nM T17569 CICM85 127031578 IC50 > 32000 nM T17569 C6AK9S 127032149 IC50 = 1200 nM T17569 CMB2T5 127032150 IC50 = 600 nM T17569 C9R4SO 127032151 IC50 = 1200 nM T17569 COK4D6 135401985 IC50 = 67 nM T17569 C7L1SH 135401986 IC50 = 130 nM T17569 C1DM3K 135401987 IC50 = 130 nM T17569 CM5JV9 135402002 IC50 = 262 nM T17569 C73STU 135402003 IC50 = 34 nM T17569 CT0JS4 135433132 IC50 = 100 nM T17569 CWU8B0 135443450 IC50 = 490 nM T17569 CQ5A3W 135450037 IC50 = 190 nM T17569 C1PA5R 135450069 IC50 = 85 nM T17569 C9L6WN 135450097 IC50 = 120 nM T17569 CDF6O0 135450098 IC50 = 280 nM T17569 CQ2RN7 135450099 IC50 = 140 nM T17569 CO23BP 135453443 IC50 = 540 nM T17569 CS3IU4 135528474 IC50 = 124 nM T17569 CP8T7X 135532460 IC50 = 90 nM T17569 C7GT2D 135532473 IC50 = 170 nM T17569 CR1O0X 135532763 IC50 = 70 nM T17569 CJB6D5 135532777 IC50 = 160 nM T17569 CIW9S8 135532890 IC50 = 149 nM T17569 CGD20L 135532893 IC50 = 160 nM T17569 C7ORW1 135547867 IC50 = 159 nM T17569 CZD1G5 135547981 IC50 = 419 nM T17569 CJZV93 135843671 IC50 = 70 nM T17569 C8SF0Y 135843672 IC50 = 30 nM T17569 C52NZK 135843695 IC50 = 310 nM T17569 CZ24TR 135843701 IC50 = 190 nM T17569 CLAY68 135843720 IC50 > 1000 nM T17569 CPO46U 135843728 IC50 = 75 nM T17569 CEJX68 135843730 IC50 > 1000 nM T17569 CX07SO 135843731 IC50 > 1000 nM T17569 CDV73T 135843739 IC50 = 580 nM T17569 CZ31NJ 135843751 IC50 = 15 nM T17569 CKZ20B 135843758 IC50 = 440 nM T17569 CI5XS8 135843764 IC50 = 440 nM T17569 CX0D8E 135843766 IC50 = 310 nM T17569 CR49PV 135843788 IC50 = 820 nM T17569 C47QCR 135843801 IC50 = 48 nM T17569 CWCR58 135843817 IC50 = 660 nM T17569 CW0SE1 135843822 IC50 > 1000 nM T17569 C14MLR 135843840 IC50 = 150 nM T17569 CU9T1A 135843881 IC50 = 660 nM T17569 C5XMC4 135843887 IC50 = 150 nM T17569 C9Q2XW 135843919 IC50 = 590 nM T17569 CGOD08 135843966 IC50 = 750 nM T17569 CO39WP 135843968 IC50 = 420 nM T17569 C46LJO 135843975 IC50 = 440 nM T17569 CJ2YG6 135843976 IC50 = 230 nM T17569 C2FCA6 135843981 IC50 = 160 nM T17569 CCW75G 135843988 IC50 = 510 nM T17569 C2UZ3F 135843992 IC50 = 57 nM T17569 CS7D2C 135843993 IC50 = 94 nM T17569 C9O1FT 135843995 IC50 = 740 nM T17569 CERB64 135844010 IC50 = 650 nM T17569 C1Y4ME 135844017 IC50 = 200 nM T17569 C8P0RS 135844066 IC50 = 970 nM T17569 CKVL36 135960821 IC50 > 1000 nM T17569 CT74UB 135960822 IC50 = 200 nM T17569 CM31KA 135967831 IC50 = 5600 nM T17569 C4YI3G 135967841 IC50 = 280 nM T17569 CKZL60 135967842 IC50 = 750 nM T17569 C2EFY0 135967846 IC50 = 200 nM T17569 C59OMK 135967850 IC50 = 350 nM T17569 C8BI4Z 135967861 IC50 = 275 nM T17569 CEH71P 135967866 IC50 = 440 nM T17569 CXL97Q 135967871 IC50 = 370 nM T17569 C57KQJ 135967876 IC50 = 547 nM T17569 C1MDS0 137028323 IC50 = 34 nM T17569 C3O6RT 137028324 IC50 = 65 nM T17569 CLF0O8 137028325 IC50 = 170 nM T17569 CI9NJ2 137028326 IC50 = 89 nM T17569 CRS69O 137028327 IC50 = 92 nM T17569 C5ZEO8 137028328 IC50 > 10000 nM T17569 C81HDS 137028329 IC50 > 10000 nM T17569 CC5I2A 137028330 IC50 > 10000 nM T17569 C39KJY 137028331 IC50 = 30 nM T17569 CBQW73 137028332 IC50 > 10000 nM T17569 C0S5WZ 137028333 IC50 > 10000 nM T17569 C49SOG 137028334 IC50 = 55 nM T17569 CICJ40 137028335 IC50 > 10000 nM T17569 CG64SP 137028336 IC50 = 52 nM T17569 CV57BS 137028337 IC50 = 28 nM T17569 C6P0UB 137028338 IC50 = 60 nM T17569 CUT6O2 137028352 IC50 > 10000 nM T17569 CTY35E 137028353 IC50 = 52 nM T17569 CXS17K 137028354 IC50 = 47 nM T17569 C6IQB8 137028355 IC50 = 32 nM T17569 CJLB61 137633993 IC50 = 62 nM T17569 C4B7UM 137640060 IC50 = 137 nM T17569 CVLN62 137640626 IC50 = 233 nM T17569 CY98CE 137642361 IC50 = 283 nM T17569 CUMA78 137644191 IC50 = 56 nM T17569 CY1HN6 137645732 IC50 = 148 nM T17569 CFPE40 137646880 IC50 = 161 nM T17569 C4O0JE 137647028 IC50 = 195 nM T17569 C6KR7G 137651362 IC50 > 10000 nM T17569 CANL61 137651426 IC50 = 290 nM T17569 CZ2MT3 137652584 IC50 = 116 nM T17569 C0O5HF 137654037 IC50 = 276 nM T17569 CA7B5Z 137656105 IC50 = 84 nM T17569 COH35U 137657930 IC50 = 26 nM T17569 CY07GS 137662191 IC50 = 153 nM T17569 CW9P6A 145964460 IC50 > 30000 nM T17569 CQR49Z 145965116 IC50 > 30000 nM T17569 CR6L2G 145967358 IC50 > 30000 nM T17569 CHXE25 145978207 IC50 > 30000 nM T17569 CXW4J6 155512369 IC50 = 3200 nM T17569 CG73TZ 155513551 IC50 = 2200 nM T17569 COB5Q1 155522288 IC50 = 260 nM T17569 CKOX20 155523419 IC50 = 2700 nM T17569 C3D0OJ 155531897 IC50 = 10000 nM T17569 CSZ8V9 155533317 IC50 = 4800 nM T17569 C8Q4KS 155537210 IC50 = 5600 nM T17569 CG8I5F 155538033 IC50 = 60 nM T17569 C6KX1G 155538348 IC50 = 220 nM T17569 C1LPN9 155540433 IC50 = 2100 nM T17569 CI0GS3 155545394 IC50 = 4800 nM T17569 CG07WS 155547154 IC50 = 1400 nM T17569 CON20B 155550001 IC50 = 3400 nM T17569 D00UCP 7824621 IC50 = 6700 nM T17569 D00WKK 11710246 IC50 = 256 nM T17569 D06BMZ 46885513 IC50 = 204 nM T17569 D07VWP 656730 IC50 = 700 nM T17569 D08BMM 6312649 IC50 = 16000 nM T17569 D08LZZ 21678144 IC50 = 500 nM T17569 D0A5KP 11588169 IC50 = 2869 nM T17569 D0D8JU 46885546 IC50 = 7107 nM T17569 D0I2NX 3545567 IC50 = 4100 nM T17569 D0J0OY 44418147 IC50 = 997 nM T17569 D0K7RO 11646379 IC50 = 3357 nM T17569 D0R5OF 46885515 IC50 = 3242 nM T17569 D0R9CF 11302540 IC50 = 3450 nM T17569 D0XB2Z 44418200 IC50 = 924 nM T17569 D0Y8AB 46885586 IC50 = 16390 nM T95605 D0G0TS 119192 Ki = 418 nM T95605 C7A3EH 1230851 EC50 > 80000 nM T95605 CA1Y2P 1230852 EC50 > 80000 nM T95605 C7L1HF 1920221 EC50 > 80000 nM T95605 C4G9CE 1941471 EC50 > 80000 nM T95605 C3P9EW 1951822 EC50 > 80000 nM T95605 C20LJC 4679731 EC50 > 80000 nM T95605 CQR16D 10339735 EC50 > 80000 nM T95605 CO47VD 11657884 IC50 = 11.1 nM T95605 C9KCA5 24868215 IC50 = 0.95 nM T95605 CFP9S1 44157038 EC50 > 80000 nM T95605 CS64NI 44354075 IC50 = 0.7 nM T95605 CWJX37 44354085 IC50 = 2.8 nM T95605 C0J9UW 44354086 IC50 = 0.23 nM T95605 C5Y7PD 44354087 IC50 = 0.78 nM T95605 COFV37 44354088 IC50 = 0.3 nM T95605 C5F9XB 44354111 IC50 = 4 nM T95605 CP9TU5 44354112 IC50 = 6.9 nM T95605 CE7C0O 44354113 IC50 = 3.5 nM T95605 C3LE1I 44354120 IC50 = 0.9 nM T95605 C3SAZ7 44354121 IC50 = 500 nM T95605 CR82IU 44354154 IC50 = 5.3 nM T95605 CJL69G 44354211 IC50 = 3.1 nM T95605 C51YEP 44354212 IC50 = 1.8 nM T95605 CTW49H 44354244 IC50 = 0.67 nM T95605 C96DTU 44354245 IC50 = 2.1 nM T95605 C7UL8I 44354302 IC50 = 5.1 nM T95605 C39YIP 44354303 IC50 = 3.5 nM T95605 CH8W9B 44354304 IC50 = 3 nM T95605 CU0SY5 44354305 IC50 = 3.2 nM T95605 CNK7H5 44363934 IC50 = 2.7 nM T95605 C2H1UE 44384829 Ki = 63 nM T95605 CWI8C2 44447826 Ki = 210 nM T95605 C1KIX8 44447828 Ki = 17 nM T95605 CVH63S 44447863 Ki = 0.74 nM T95605 C3UE1C 44447864 Ki = 21 nM T95605 C34DVM 44447865 Ki = 1000 nM T95605 CJ50IK 45102614 Ki = 8.8 nM T95605 CF63HL 49798969 EC50 = 54.2 nM T95605 CX9M3E 49837912 EC50 > 80000 nM T95605 CVQM43 51035368 EC50 > 80000 nM T95605 C65GEF 51035373 EC50 > 80000 nM T95605 C9YIZ5 52914819 EC50 > 80000 nM T95605 C6S9YI 52914822 EC50 > 80000 nM T95605 C3Y4DQ 52914826 EC50 > 80000 nM T95605 C9FJ6G 52951375 Ki = 38 nM T95605 CL1E9Q 52951376 Ki = 20 nM T95605 C2LOM8 52951377 Ki = 100 nM T95605 CS3U7Z 52951476 Ki = 6.7 nM T95605 C0XZ2V 52951477 Ki = 4.4 nM T95605 CNI2F4 52951478 Ki = 4.3 nM T95605 CC4U3O 53245521 EC50 > 80000 nM T95605 C3WTY4 53245542 EC50 > 80000 nM T95605 CE7A9B 53245571 EC50 > 80000 nM T95605 CH4EO6 53245574 EC50 > 80000 nM T95605 CMJ62D 53245590 EC50 > 80000 nM T95605 CQHV82 53245615 EC50 > 80000 nM T95605 C69HCK 53245626 EC50 > 80000 nM T95605 CNFI86 54580106 Ki = 5.4 nM T95605 CPO5M6 54580107 Ki = 51 nM T95605 C6ZX1P 54580108 Ki = 3700 nM T95605 CYJ93A 54581089 Ki = 140 nM T95605 CP92RB 54582126 Ki = 0.61 nM T95605 CX7K3E 54582127 Ki = 16 nM T95605 CX90US 54583072 Ki = 63 nM T95605 CDXP96 54583073 Ki = 590 nM T95605 C2SCE8 54583074 Ki = 690 nM T95605 CSN46R 54583075 Ki = 25 nM T95605 CCY5W1 54583076 Ki = 1600 nM T95605 CHSI63 54585021 Ki = 24 nM T95605 CHNT83 54585022 Ki = 83 nM T95605 C24YLS 54585023 Ki = 44 nM T95605 C9I4DC 54585988 Ki = 56 nM T95605 CO0P4Z 54585989 Ki = 1300 nM T95605 CUQX42 54585990 Ki = 5.4 nM T95605 C0HI5E 54758538 EC50 > 80000 nM T95605 CZ63WS 54758539 EC50 > 80000 nM T95605 CC6F4U 56593272 EC50 > 80000 nM T95605 CY5VX7 56593273 EC50 > 80000 nM T95605 C1RJX8 56593274 EC50 > 80000 nM T95605 CX1N3I 56593278 EC50 > 80000 nM T95605 CMF4H8 56593279 EC50 > 80000 nM T95605 CB75SU 56593281 EC50 > 80000 nM T95605 C2J7VC 56593282 EC50 > 80000 nM T95605 CA9OV0 56593283 EC50 > 80000 nM T95605 C2FHP7 56593284 EC50 > 80000 nM T95605 CNG48L 56593288 EC50 > 80000 nM T95605 CY1N5C 56593289 EC50 > 80000 nM T95605 C7ZL2B 56593290 EC50 > 80000 nM T95605 CD06NY 56593291 EC50 > 80000 nM T95605 CQ60KY 56593292 EC50 > 80000 nM T95605 CNB83L 56593293 EC50 > 80000 nM T95605 CCG58A 72737612 Ki = 69 nM T95605 CG62IS 73346308 EC50 > 80000 nM T95605 CU83RW 73346899 Ki = 330 nM T95605 CO8S0I 73347807 EC50 > 80000 nM T95605 CH2YN5 73349346 EC50 > 80000 nM T95605 C6V7YB 73350917 EC50 > 80000 nM T95605 C8PZ4T 73352405 EC50 > 80000 nM T95605 C4G6FB 73353870 EC50 > 80000 nM T95605 C5IVA1 73355398 EC50 > 80000 nM T95605 CGTQ84 73356947 EC50 > 80000 nM T95605 CQ91AR 73356948 EC50 > 80000 nM T95605 C2BZA6 101171051 IC50 = 21.2 nM T95605 C9O6WP 122192055 IC50 = 405 nM T95605 C1DSL0 122192056 IC50 = 0.26 nM T95605 C3KWU5 122192057 IC50 = 28.9 nM T95605 C98IKC 122192058 IC50 = 1425 nM T95605 C0A5VN 122192059 IC50 = 29.7 nM T95605 CVZT87 127032101 Ki = 0.74 nM T95605 CCLG54 127032411 Ki = 2.5 nM T95605 C1GA4W 132547200 Ki = 700 nM T95605 CW7V8Q 134134595 Ki = 500 nM T95605 CIZ1T2 134136231 Ki = 2030 nM T95605 C07SHR 134138287 Ki = 11000 nM T95605 C8NFR1 134140868 Ki = 227 nM T95605 CE5Z0K 134142369 Ki = 147 nM T95605 C3S9GD 134143837 Ki = 1430 nM T95605 CK03XR 134144300 Ki = 110 nM T95605 CMGT90 134145547 Ki = 12 nM T95605 C2KR6X 134145567 Ki = 615 nM T95605 CHR4S3 134146201 Ki = 6000 nM T95605 CO8Q7F 134147225 Ki = 873 nM T95605 CRH73L 134152554 Ki = 69 nM T95605 CKS0C3 134153118 Ki = 29 nM T95605 C87ZMF 134155365 Ki = 12 nM T95605 C2MKS7 137645783 Ki = 1600 nM T95605 CY6N5R 137646112 Ki = 261.8 nM T95605 COX29R 137651580 Ki = 4200 nM T95605 CN74UT 137651867 Ki = 474.1 nM T95605 CLF01S 137656771 Ki = 619.5 nM T95605 CVP06T 137660279 Ki = 67 nM T95605 CAH73J 155525403 Ki = 3.981 nM T95605 CY8XR1 155547077 Ki = 0.955 nM T95605 CYX16L 155548706 Ki = 3.467 nM T95605 C2SA8V 155559775 Ki = 1.202 nM T95605 CY4IX3 155569268 Ki = 7.244 nM T95605 D00TPV 5311318 Ki = 0.7413 nM T95605 D0H8AI 25077406 Ki = 4.9 nM T95605 D0OJ7S 5311451 Ki = 74 nM T52624 D0B0AX 5328127 IC50 > 50000 nM T52624 D0OB0F 5328940 IC50 = 4000 nM T52624 D0VF6E 1401 IC50 = 17000 nM T52624 D0H8KG 5311382 IC50 = 6.5 nM T52624 CE1US5 652633 IC50 > 10000 nM T52624 C3P8CG 5327885 IC50 = 1 nM T52624 CYRW80 5327889 IC50 = 680 nM T52624 CLH9Y3 5327908 IC50 = 1 nM T52624 C04BUF 5327909 IC50 = 1 nM T52624 CPT61U 5328112 IC50 = 1110 nM T52624 CXR9K1 5328115 IC50 = 660 nM T52624 CM0H5O 5328117 IC50 = 340 nM T52624 CDM98R 5328125 IC50 > 50000 nM T52624 CDY2O3 5328134 IC50 = 240 nM T52624 CC1O0M 5328135 IC50 = 450 nM T52624 C14LVT 5328137 IC50 = 1200 nM T52624 COT45A 5328149 IC50 = 270 nM T52624 C5EN6O 5328163 IC50 = 370 nM T52624 C0Z8KJ 5328458 IC50 > 10000 nM T52624 C10RHA 5328469 IC50 = 150 nM T52624 CJM61R 5328509 IC50 = 790 nM T52624 CCZ0J4 5328642 IC50 = 54 nM T52624 C0AY2D 5328647 IC50 = 4.6 nM T52624 C91NVI 5328648 IC50 > 25 nM T52624 CR0PI3 5328649 IC50 = 3 nM T52624 CART86 5328650 IC50 = 58 nM T52624 CWX63A 5329004 IC50 = 3400 nM T52624 CSY10K 5329111 IC50 = 4670 nM T52624 CBS40G 5330125 IC50 = 9100 nM T52624 CNWK81 5330126 IC50 = 7500 nM T52624 CV7GX5 5330127 IC50 = 1800 nM T52624 CWAR90 5330128 IC50 = 4000 nM T52624 CDG3Z1 5330129 IC50 = 2700 nM T52624 C09VSN 5330130 IC50 = 1300 nM T52624 CNMJ73 5330131 IC50 = 5900 nM T52624 CV4U8Y 5330132 IC50 = 3500 nM T52624 C6D7WJ 5330133 IC50 = 2100 nM T52624 C2UX4V 5330134 IC50 = 2900 nM T52624 CH38FW 5330135 IC50 = 980 nM T52624 CWQ47D 5330136 IC50 = 1500 nM T52624 CLI47K 5330157 IC50 = 1800 nM T52624 CNI15R 5330158 IC50 = 1200 nM T52624 C4IA7N 5330159 IC50 = 3400 nM T52624 CW8G9J 5330166 IC50 = 12000 nM T52624 C7Z2YH 5330167 IC50 = 7900 nM T52624 CEX9A7 5330168 IC50 > 25000 nM T52624 C3I6KF 5330169 IC50 = 11000 nM T52624 COB2X8 10602350 IC50 = 4300 nM T52624 CJO8Q1 10738332 IC50 = 1300 nM T52624 D00YCU 667662 IC50 = 130 nM T52624 D01FWD 606669 IC50 = 2300 nM T52624 D01MUN 5328453 IC50 = 2000 nM T52624 D02XKJ 5328466 IC50 = 1900 nM T52624 D0K2YG 5328512 IC50 = 1360 nM T90682 CU3EJ0 96215 EC50 = 3000 nM T90682 C58SGV 1502041 EC50 = 17500 nM T90682 C5RM2I 5310987 EC50 = 400 nM T90682 CA8CU6 10103145 EC50 = 101000 nM T90682 D0O9UH 6603697 EC50 = 70000 nM T90682 D0U4HM 5521 IC50 = 22090 nM T07740 C0I8GC 14985965 IC50 > 100000 nM T07740 C0NI3L 51003771 IC50 = 24000 nM T07740 C3XQE2 52337837 IC50 > 100000 nM T07740 C4E1NK 57331209 IC50 > 50000 nM T07740 CGUA26 57331668 IC50 > 50000 nM T07740 CM1G2P 59568656 IC50 > 50000 nM T25861 D06XDJ 2782 IC50 = 9100 nM T25861 C6PU5E 270291 IC50 > 100000 nM T25861 C4HQ7V 284016 IC50 = 48600 nM T25861 CZN6S9 743974 EC50 > 50118.72 nM T25861 C6EM0S 1096735 IC50 = 1260 nM T25861 C5E4RY 1096815 IC50 = 630 nM T25861 C5ADZ4 4519833 IC50 = 800 nM T25861 CZXR85 4871557 IC50 = 30400 nM T25861 CX31PA 4915642 IC50 = 19300 nM T25861 CUZC83 5308428 EC50 = 450 nM T25861 CNG21Y 6991896 IC50 > 100000 nM T25861 CT1HK3 10598093 IC50 = 18460 nM T25861 CY7O0L 53378752 IC50 = 282 nM T25861 CNQ51P 53475435 IC50 = 720 nM T25861 C09LTC 56944680 IC50 = 500 nM T25861 CPUM70 59740711 IC50 > 100000 nM T25861 COT21H 71723590 IC50 > 100000 nM T25861 CT29AF 71818278 IC50 = 800 nM T25861 CNQ38C 71818279 IC50 = 6300 nM T25861 C7APU4 71818280 IC50 = 1600 nM T25861 C61GSX 71818281 IC50 = 400 nM T25861 C23DTZ 71818282 IC50 = 800 nM T25861 CQ20DY 71818427 IC50 = 12600 nM T25861 C5GI1E 71818428 IC50 > 25000 nM T25861 CK1I7A 71818429 IC50 = 2500 nM T25861 CH51FU 71818430 IC50 = 6300 nM T25861 CW20HQ 71818431 IC50 = 250 nM T25861 CDIR63 71818432 IC50 = 80 nM T25861 C9K3HJ 71818433 IC50 = 160 nM T25861 CFQ9C5 71818573 IC50 = 32 nM T25861 CE4K3S 71818574 IC50 = 250 nM T25861 C2L7TX 71818575 IC50 = 100 nM T25861 CPFB17 71818576 IC50 = 1000 nM T25861 CHFG76 71818577 IC50 = 316 nM T25861 CEH0X1 71818578 IC50 = 316 nM T25861 C4H6ZC 71818579 IC50 = 10000 nM T25861 CN3C5I 71818710 IC50 = 20000 nM T25861 CS13DM 121277209 EC50 = 138 nM T25861 C9C5BR 121277212 EC50 = 236 nM T25861 CV83UW 121279842 EC50 = 19 nM T25861 CEK6B1 139300630 IC50 > 10000 nM T25861 D03LVL 53464483 IC50 > 25000 nM T25861 D0JV2P 2455 IC50 = 4210 nM T25861 D0T7GC 56964346 IC50 = 540 nM T96892 D02XNW 5494449 IC50 = 420 nM T96892 D03HUX 49792852 IC50 = 744 nM T96892 D04UUD 10430360 IC50 = 340 nM T96892 D05PZB 135398495 IC50 = 685 nM T96892 D08FIX 135398499 IC50 = 0.41 nM T96892 D0E3TC 44259 IC50 = 0.542 nM T96892 D0O0LS 25141092 IC50 > 10000 nM T96892 C4DW3Y 660621 IC50 = 1185 nM T96892 C3GHQ1 690227 IC50 > 5000 nM T96892 CIZ9D2 2216908 IC50 > 5000 nM T96892 CJAQ19 2491127 IC50 = 388 nM T96892 C1OW6X 3141330 IC50 > 5000 nM T96892 CF7HW1 3620985 IC50 = 400 nM T96892 CA3C5S 3685259 IC50 = 180 nM T96892 CB7WK3 5938113 IC50 = 1400 nM T96892 CV50PJ 12451684 IC50 = 6100 nM T96892 CJ8W9Z 16044323 IC50 > 5000 nM T96892 C3P8XU 16760499 IC50 = 440 nM T96892 C46DEZ 17816913 IC50 > 20000 nM T96892 CRAH02 42647778 IC50 > 5000 nM T96892 C9WL5N 42647801 IC50 > 5000 nM T96892 CBI04W 42647935 IC50 = 1116 nM T96892 CSP6D8 43831079 IC50 = 4126 nM T96892 C1U7PZ 43831080 IC50 = 1774 nM T96892 C3VRO9 44557921 IC50 > 10000 nM T96892 CLS29B 46872626 IC50 > 10000 nM T96892 C6J4OP 47001335 IC50 = 192 nM T96892 CF91RS 49843531 IC50 > 10000 nM T96892 C2Y6QS 50938552 IC50 > 10000 nM T96892 C9NYP4 51036677 IC50 > 10000 nM T96892 C4WRY3 51037112 IC50 > 10000 nM T96892 CRI28Z 51037948 IC50 > 10000 nM T96892 CV13QY 58540422 IC50 > 10000 nM T96892 CMO15Y 63901349 IC50 = 160000 nM T96892 CV63UL 67240318 IC50 > 10000 nM T96892 CCN01X 71547862 IC50 > 10000 nM T96892 C6R8DI 72943374 IC50 = 258 nM T96892 C4U5NV 73442760 IC50 = 37 nM T96892 CGDB30 74538658 IC50 = 19 nM T96892 CGJ0Q3 78350436 IC50 = 2100 nM T96892 C27SIH 78350438 IC50 = 31000 nM T96892 CGKW40 78350469 IC50 = 3100 nM T96892 C6FR9J 78350471 IC50 = 4200 nM T96892 CS4A3I 78673829 IC50 = 1000 nM T96892 C7QSR8 85325330 IC50 = 520 nM T96892 C0NR6S 85325332 IC50 = 650 nM T96892 CY0UC4 90645194 IC50 > 10000 nM T96892 CY7BI2 118706214 IC50 > 10000 nM T96892 C6S4XB 118720606 IC50 = 410 nM T96892 C2K6LE 118720607 IC50 = 24000 nM T96892 C06LWS 118720608 IC50 = 5100 nM T96892 CS4I7U 118720609 IC50 = 7.6 nM T96892 C75PHN 119058124 IC50 = 2 nM T96892 CJ6FQ7 119058125 IC50 = 410 nM T96892 CWDX84 119058126 IC50 = 13 nM T96892 C5YJ9E 122705889 IC50 = 900 nM T96892 CS2E6X 127048234 IC50 = 5000 nM T96892 C2YHT0 127048915 IC50 = 670 nM T96892 CF0KU7 127050847 IC50 = 520 nM T96892 C24DQX 127051101 IC50 = 64 nM T96892 CH1YA6 127051102 IC50 = 80 nM T96892 C1Y2GO 127051103 IC50 = 1 nM T96892 CP73XR 127051104 IC50 = 25 nM T96892 CCZH52 127051105 IC50 = 260 nM T96892 C6LNW2 127052230 IC50 = 4 nM T96892 CR48OV 127052231 IC50 = 36 nM T96892 CS59XH 127052232 IC50 = 210 nM T96892 CW8Z6C 127052233 IC50 = 0.3 nM T96892 C2AN7T 134611886 IC50 > 100000 nM T96892 CJI0G1 135520135 IC50 = 2800 nM T96892 CHA4N2 136013680 IC50 > 10 nM T96892 CH64ID 136175114 IC50 > 10000 nM T96892 C1YUD0 136219394 IC50 > 10 nM T96892 COG2M5 136242661 Ki = 0.47 nM T96892 CIU8W3 136254389 IC50 > 10 nM T96892 CSGM03 137210056 IC50 = 1000 nM T96892 C04YDK 137248544 Ki = 0.39 nM T96892 C2J5CN 137293686 Ki = 2.3 nM T96892 C97CMT 137293687 Ki = 358 nM T96892 CDB68K 137293702 Ki > 650 nM T96892 CRYI28 137293705 Ki = 3.1 nM T96892 CMB78I 137301774 Ki = 0.68 nM T96892 CHF1V3 137301775 Ki = 46 nM T96892 C0W3KM 137631515 IC50 = 120 nM T96892 C2Z6PU 137632011 IC50 = 3500 nM T96892 C6VKD9 137633401 IC50 = 9.2 nM T96892 CU75HC 137633476 IC50 = 3700 nM T96892 CT41DA 137636064 IC50 = 400 nM T96892 CYH3P1 137636760 IC50 = 6800 nM T96892 CFYB36 137638498 Ki = 8.8 nM T96892 CGP48Y 137639114 IC50 = 1.5 nM T96892 CNU81W 137641500 IC50 = 8.8 nM T96892 C6G5BQ 137642064 IC50 = 8900 nM T96892 CJ4MI7 137642078 IC50 = 1.1 nM T96892 CZ3C1M 137643225 IC50 = 720 nM T96892 CINF50 137644022 IC50 = 2600 nM T96892 C4U9QF 137646381 IC50 = 1300 nM T96892 CMZ02P 137649794 IC50 = 0.15 nM T96892 C1KO7R 137651632 IC50 = 2100 nM T96892 CP04RX 137652802 IC50 = 740 nM T96892 C5MG7R 137653946 IC50 = 1.5 nM T96892 CM9H2O 137655933 IC50 = 12 nM T96892 C40GAX 137659707 IC50 = 7700 nM T96892 CR2OA8 155510507 IC50 = 141 nM T96892 C2MD1Q 155513187 IC50 > 10000 nM T96892 C2WGR6 155518450 IC50 > 5000 nM T96892 CZ3RW5 155521164 IC50 = 112 nM T96892 CTXD61 155522409 IC50 = 222 nM T96892 C01QHJ 155522952 IC50 = 122 nM T96892 CP8A0W 155523587 IC50 = 599 nM T96892 CHQ63Z 155531664 IC50 = 638 nM T96892 C8OL9Y 155532496 IC50 = 1701 nM T96892 C0AR4Z 155533016 IC50 > 5000 nM T96892 CDZ18P 155535001 IC50 = 241 nM T96892 CR9G3K 155538487 IC50 = 540 nM T96892 CB01CY 155540962 IC50 = 707 nM T96892 CAYF68 155543222 IC50 = 269 nM T96892 C1KBH2 155547976 IC50 = 350 nM T96892 C19QDP 155549136 IC50 = 575 nM T96892 C0STI2 155549197 IC50 > 5000 nM T96892 CH3K7T 155552256 IC50 > 5000 nM T96892 CHE7F8 155554129 IC50 = 1417 nM T96892 CN4TI9 155555255 IC50 = 98 nM T96892 CHU10X 155558521 IC50 > 5000 nM T96892 CE4LF2 155558943 IC50 = 313 nM T96892 CG4HQ6 155559449 IC50 > 5000 nM T96892 CUW59T 155559912 IC50 = 1353 nM T96892 CT5W1V 155566733 IC50 = 494 nM T96892 D05GMB 135461425 Ki = 149 nM T96892 D09HVH 135566652 IC50 > 10 nM T96892 D09LPL 5329103 IC50 = 760 nM T96892 D0IR6U 5494425 IC50 = 330 nM T92076 D03YGR 156419 EC50 = 80 nM T92076 D04CJE 44201334 IC50 = 1.4 nM T92076 D0H8OA 46917559 IC50 = 12 nM T92076 D0R7IU 9910902 IC50 = 73 nM T92076 D02FEA 3336 EC50 = 1000 nM T92076 D03XIS 158796 EC50 = 80 nM T92076 D07XPT 10345214 IC50 = 146 nM T92076 D0G1RH 6918446 IC50 = 0.003 nM T92076 C5C2BD 156418 EC50 = 19.95 nM T92076 CNZ6O8 158797 EC50 = 80 nM T92076 C9T4KC 671770 IC50 > 30000 nM T92076 CX32UY 1547139 IC50 > 30000 nM T92076 CR1M9X 3123058 IC50 > 10000 nM T92076 CW5B1T 3431830 EC50 = 4000 nM T92076 C5ZOR1 3781744 EC50 = 2000 nM T92076 C5MZE2 4341046 EC50 = 4000 nM T92076 CT7PY1 4564558 EC50 = 4000 nM T92076 CF41RA 7145229 EC50 = 1200 nM T92076 CTN56U 9802994 IC50 = 68 nM T92076 CN9YD5 9868131 IC50 = 3 nM T92076 CFRS47 9910748 IC50 = 18 nM T92076 C10VOI 9930235 IC50 = 70 nM T92076 CMI58L 9956563 IC50 = 0.003 nM T92076 C25ZDX 10020257 IC50 = 2800 nM T92076 CAS6K3 10028311 IC50 = 0.4 nM T92076 CB63ML 10094574 IC50 = 140 nM T92076 CQG2L0 10109178 IC50 = 9 nM T92076 CXMV78 10111057 IC50 = 170 nM T92076 CWC98Q 10111740 IC50 = 160 nM T92076 C3H9XW 10113741 IC50 = 41 nM T92076 C5ZL9F 10115992 IC50 = 7.3 nM T92076 C4LNZ0 10120467 IC50 = 2.4 nM T92076 C3BJI2 10133274 IC50 = 180 nM T92076 CV1OS7 10135815 IC50 = 70 nM T92076 C2EYN5 10158373 IC50 = 4.4 nM T92076 C98NUM 10161939 IC50 = 520 nM T92076 CW5U2S 10180249 IC50 = 37 nM T92076 CG62JR 10210971 IC50 = 13 nM T92076 C9LRC0 10222076 IC50 = 200 nM T92076 CFI09T 10272812 IC50 = 120 nM T92076 C1NH7S 10341785 EC50 = 23 nM T92076 CBP2M4 10366358 IC50 = 790 nM T92076 CD8KU7 10387815 IC50 = 190 nM T92076 C1W4HL 10408861 EC50 = 37 nM T92076 CB9PH2 10453544 EC50 = 160 nM T92076 C1N4EP 11155912 IC50 = 14 nM T92076 C7QJW8 11191770 IC50 = 6 nM T92076 C6FR9A 11203324 IC50 = 60 nM T92076 CO89GP 11214076 IC50 = 15 nM T92076 CED23Y 11281119 IC50 = 22 nM T92076 CZ4I3R 11307362 IC50 = 70 nM T92076 CXGF34 11328907 IC50 = 11 nM T92076 CKE5W1 11384835 IC50 = 25 nM T92076 CY96UR 11398805 IC50 = 5 nM T92076 C1COT8 11408302 IC50 = 24 nM T92076 CCN39M 11410354 IC50 = 76 nM T92076 C2A7HJ 11427732 IC50 = 210 nM T92076 C03NGT 11430368 IC50 = 190 nM T92076 CP3D2O 11442305 IC50 = 13 nM T92076 CG0M5T 11451283 IC50 = 70 nM T92076 CN6PE7 11462501 IC50 = 50 nM T92076 CZD3E4 11477141 IC50 = 60 nM T92076 C9OIF7 11478504 IC50 = 150 nM T92076 CB94DA 11486852 IC50 = 190 nM T92076 CXHN40 11488770 IC50 = 5 nM T92076 C1KVI8 11545487 EC50 = 27 nM T92076 CH7E2Y 11706057 EC50 = 12.59 nM T92076 CWY09Q 11775322 IC50 = 1000 nM T92076 CJ52NB 11786197 IC50 = 43 nM T92076 CIT4B3 11955172 EC50 = 60 nM T92076 COS92H 11955187 EC50 = 40 nM T92076 CYHS93 11955188 EC50 = 30 nM T92076 CH95TQ 11955189 EC50 = 20 nM T92076 CGD59H 11955191 EC50 = 20 nM T92076 CWR5V2 11955209 EC50 = 36 nM T92076 CUTJ93 11955290 EC50 = 16 nM T92076 C1SZ7K 12898539 IC50 > 30000 nM T92076 CQ1Y8G 15461660 IC50 = 2300 nM T92076 CKJX89 16112870 EC50 = 60 nM T92076 C5TY4N 16735042 EC50 = 200 nM T92076 CNBR46 16735043 EC50 = 200 nM T92076 C9M8UJ 16735045 EC50 = 150 nM T92076 CZ37BS 16735429 EC50 = 400 nM T92076 C4CJM1 16735430 EC50 = 1000 nM T92076 CAP38F 16735431 EC50 = 300 nM T92076 CT2EG5 16735684 EC50 = 200 nM T92076 CS75CQ 16735877 EC50 = 400 nM T92076 CCT1F7 16736322 EC50 = 150 nM T92076 CW74OP 16736324 EC50 = 150 nM T92076 CY3BL5 16736327 EC50 = 60 nM T92076 C5XHS6 16737126 EC50 = 800 nM T92076 CXG41J 16737131 EC50 = 400 nM T92076 CJY1F4 16737152 EC50 = 150 nM T92076 C46PDI 16737168 EC50 = 150 nM T92076 C04SGF 16737306 EC50 = 800 nM T92076 CM49NK 16737307 EC50 = 2000 nM T92076 CDG6V3 16737311 EC50 = 200 nM T92076 C7I1AF 16737501 EC50 = 300 nM T92076 CO41JZ 16737642 EC50 = 800 nM T92076 C9BI3A 16737652 EC50 = 350 nM T92076 CZGT79 16737653 EC50 = 1000 nM T92076 C3K6QN 16737665 EC50 = 300 nM T92076 C2I4ZH 16737826 EC50 = 550 nM T92076 CP30VS 16737828 EC50 = 130 nM T92076 CX5WM4 16737832 EC50 = 200 nM T92076 COS30P 16737836 EC50 = 400 nM T92076 CS8PK9 16737981 EC50 = 300 nM T92076 CNUB69 16737985 EC50 = 400 nM T92076 CP69UW 16738376 EC50 = 100 nM T92076 CO2GD5 18459606 IC50 = 1000 nM T92076 CWJ7K6 19360455 IC50 = 200 nM T92076 C9JD5Y 19360456 IC50 = 140 nM T92076 C28MZO 21388140 IC50 = 11360 nM T92076 CRWY74 22640800 IC50 = 210 nM T92076 C4A1BO 22640808 IC50 = 2780 nM T92076 CKYV16 22640863 IC50 = 1000 nM T92076 CH79LM 22640903 IC50 = 10000 nM T92076 C4YO5I 22640916 IC50 = 1300 nM T92076 C4E1VF 22640930 IC50 = 3500 nM T92076 C7O8MV 22640957 IC50 = 3200 nM T92076 CY4ET8 23742117 EC50 = 6000 nM T92076 C0RK2A 23934373 EC50 = 3000 nM T92076 C2EGM8 23959728 EC50 = 15000 nM T92076 CW52OD 24753618 IC50 = 4 nM T92076 C72RCA 24753619 IC50 = 1.6 nM T92076 CYA4S0 24753707 IC50 = 2.6 nM T92076 CHM9Y0 24753709 IC50 = 4 nM T92076 CHI83W 24769038 IC50 = 0.022 nM T92076 CFA4K7 24852863 EC50 = 800 nM T92076 C9S3DZ 25175312 EC50 = 10000 nM T92076 CJ6BF9 25175471 EC50 = 2000 nM T92076 CYT3I0 25198729 IC50 = 140 nM T92076 CRXY68 25218698 IC50 = 200 nM T92076 CE6YO7 25218699 IC50 = 2200 nM T92076 C9Z5HO 25218700 IC50 = 730 nM T92076 C6C1LV 25218701 IC50 = 470 nM T92076 C7Z5RU 25218702 IC50 = 4900 nM T92076 C4SKG6 25218703 IC50 = 10000 nM T92076 CYOA85 25218704 IC50 = 3100 nM T92076 CE0T3D 25218705 IC50 = 340 nM T92076 CM1AK7 25218706 IC50 = 150 nM T92076 C6XGL0 25218707 IC50 > 30000 nM T92076 C38APB 25218708 IC50 > 30000 nM T92076 CS3VN0 25218709 IC50 = 400 nM T92076 C4TE0Q 25218710 IC50 = 1500 nM T92076 CC5O4R 25218711 IC50 = 340 nM T92076 CH6IT8 25218712 IC50 = 1000 nM T92076 C5M6ZQ 25218713 IC50 = 2800 nM T92076 CEVL92 25218714 IC50 > 30000 nM T92076 CD6Q1F 25218715 IC50 > 30000 nM T92076 CT10VR 25218716 IC50 > 30000 nM T92076 CZD6K7 25218717 IC50 > 30000 nM T92076 CDB8O4 25218718 IC50 > 30000 nM T92076 C4FPG3 25218719 IC50 > 30000 nM T92076 C3U0GI 25218720 IC50 = 2100 nM T92076 CLRP91 25218721 IC50 = 1800 nM T92076 C61EDS 25218722 IC50 > 30000 nM T92076 C1JL0B 25218723 IC50 > 30000 nM T92076 CZ8C0X 25218724 IC50 > 30000 nM T92076 CUFC42 25218725 IC50 = 18900 nM T92076 CIFX53 25218726 IC50 = 6900 nM T92076 CV57BN 25218727 IC50 > 30000 nM T92076 C1C2FD 25218728 IC50 = 360 nM T92076 C4X8GO 25218729 IC50 = 220 nM T92076 CDAT67 25218730 IC50 = 360 nM T92076 CYU62C 25218731 IC50 = 150 nM T92076 CUIH08 25218732 IC50 = 154 nM T92076 COK51L 25218733 IC50 = 1050 nM T92076 C5K8HE 25218734 IC50 = 130 nM T92076 C10LRY 25218735 IC50 = 162 nM T92076 CUN6Y4 25218736 IC50 = 197 nM T92076 C21MIL 28446917 EC50 = 3700 nM T92076 CX5D8W 28447518 EC50 = 370 nM T92076 CU3TY5 44186381 IC50 = 7000 nM T92076 CP25TZ 44186382 IC50 > 10000 nM T92076 CQGS51 44186383 IC50 > 10000 nM T92076 CRYH29 44186384 IC50 > 10000 nM T92076 C2AS7D 44186385 IC50 > 10000 nM T92076 C5DC0X 44186435 IC50 = 2300 nM T92076 C9VKS6 44186436 IC50 = 950 nM T92076 CKIP70 44186437 IC50 = 930 nM T92076 C19VMJ 44186438 IC50 = 300 nM T92076 C3QET0 44390065 IC50 > 30000 nM T92076 C6IP1J 44390115 IC50 > 30000 nM T92076 C7K3AX 44390155 IC50 > 30000 nM T92076 C13OIF 44405804 IC50 = 60 nM T92076 CA35IV 44405808 IC50 = 100 nM T92076 CR7D6F 44405809 IC50 = 600 nM T92076 C84NXZ 44405815 IC50 = 6180 nM T92076 C7Y1AR 44405839 IC50 = 440 nM T92076 CZI0A4 44405840 IC50 = 0.003 nM T92076 CZ73XV 44405841 IC50 = 6840 nM T92076 CV9N8I 44405847 IC50 = 970 nM T92076 C1BD4G 44405848 IC50 = 750 nM T92076 C4RSJ1 44405849 IC50 = 240 nM T92076 CF17ZX 44405850 IC50 = 8430 nM T92076 CA3Y5R 44405851 IC50 = 1390 nM T92076 C3D1AU 44405852 IC50 = 1270 nM T92076 CP8A1I 44405853 IC50 = 1570 nM T92076 CRX4T1 44405855 IC50 = 360 nM T92076 CGX1R3 44405856 IC50 = 340 nM T92076 CV9C8O 44405861 IC50 = 1560 nM T92076 CJV32B 44405873 IC50 = 250 nM T92076 CFU18H 44405874 IC50 = 160 nM T92076 CY7F2O 44405884 IC50 = 1000 nM T92076 C92QIO 44405885 IC50 = 1350 nM T92076 C5FAB0 44405886 IC50 = 50 nM T92076 C5E1OM 44405889 IC50 = 140 nM T92076 CY95PD 44405890 IC50 = 270 nM T92076 CG5ZP0 44405891 IC50 = 880 nM T92076 CW26CP 44405892 IC50 = 2470 nM T92076 C5TB8F 44405894 IC50 = 140 nM T92076 CQ5O9A 44405899 IC50 = 2840 nM T92076 C7JE0S 44405900 IC50 = 2670 nM T92076 C3M4OH 44405902 IC50 = 3300 nM T92076 CZW56Y 44405904 IC50 = 9430 nM T92076 C8N4RG 44405908 IC50 = 1190 nM T92076 CQ85YK 44405909 IC50 = 1160 nM T92076 CNE7F0 44405912 IC50 = 4600 nM T92076 C1C5TM 44405917 IC50 = 3860 nM T92076 CEXG45 44462802 EC50 = 23 nM T92076 CV92IJ 44541354 IC50 = 4.8 nM T92076 CW82GS 44542479 EC50 > 5000 nM T92076 C1LI4D 44542480 EC50 > 5000 nM T92076 CBX96K 44542482 EC50 = 1180 nM T92076 CH7V3F 44542629 EC50 = 148 nM T92076 C1NB6V 44542630 EC50 = 70 nM T92076 CX0PO9 44542631 EC50 > 5000 nM T92076 CHON74 44542927 EC50 > 5000 nM T92076 CS94BN 44542931 EC50 = 1580 nM T92076 CG9R1W 44543086 EC50 = 233 nM T92076 CW3F1O 44543087 EC50 = 2340 nM T92076 CT31FG 44543088 EC50 = 92 nM T92076 C9XUP8 44543243 EC50 = 41 nM T92076 C8F3XS 44543375 EC50 = 57 nM T92076 C89CGP 44543376 EC50 = 1920 nM T92076 C3L5ER 44583033 IC50 = 11 nM T92076 C1ED7Y 44610739 IC50 = 25 nM T92076 CI6D3E 45139806 IC50 > 30000 nM T92076 CZ5TB6 45139807 IC50 = 2100 nM T92076 CGD7B0 45139808 IC50 = 3300 nM T92076 C6T9NP 45139809 IC50 = 2100 nM T92076 CSR27V 45139810 IC50 = 5500 nM T92076 CD40YV 45139811 IC50 > 30000 nM T92076 CF2X8D 45140000 IC50 > 30000 nM T92076 C8PG7W 45140001 IC50 > 30000 nM T92076 CVP54L 45140003 IC50 = 15900 nM T92076 C4IJ9V 45140004 IC50 = 2200 nM T92076 C4C3SV 45140005 IC50 = 1100 nM T92076 CG4VP0 45140006 IC50 = 2700 nM T92076 C8O6FI 45140210 IC50 = 3700 nM T92076 CT3MF5 45140212 IC50 = 170 nM T92076 CIZ5Q9 45140595 IC50 = 1.6 nM T92076 CBGY18 45140596 IC50 = 4.2 nM T92076 CG64RO 45140790 IC50 = 27 nM T92076 C6RIO3 45140791 IC50 = 4.2 nM T92076 C40UQG 45140792 IC50 = 19 nM T92076 COY58K 45140793 IC50 = 12.6 nM T92076 CY7B6Q 45140794 IC50 = 1.8 nM T92076 C61FWA 45140795 IC50 = 13 nM T92076 CTF8O7 45140969 IC50 = 2.7 nM T92076 CSG41K 45140970 IC50 = 3.4 nM T92076 CW4JT2 45140971 IC50 = 460 nM T92076 COU9R7 45140972 IC50 = 520 nM T92076 C0C2HB 45140973 IC50 = 1100 nM T92076 CQ1C9I 45140974 IC50 = 2900 nM T92076 C5QRD9 45141171 IC50 = 230 nM T92076 C2GR3X 45141172 IC50 = 30 nM T92076 C4F7JS 45141173 IC50 = 120 nM T92076 C8W4LQ 45141174 IC50 = 10000 nM T92076 C45XOM 45141389 IC50 = 3.9 nM T92076 CQ23IP 45141390 IC50 = 6.6 nM T92076 CKZ81J 45141391 IC50 = 2.5 nM T92076 C48SVL 45141392 IC50 = 8.1 nM T92076 C47AYD 45484067 EC50 > 5000 nM T92076 C5SB6T 45484073 EC50 > 5000 nM T92076 C51VXD 46228785 IC50 = 1400 nM T92076 COXR81 46228881 IC50 = 6600 nM T92076 CCWK45 46871629 IC50 = 23 nM T92076 CKUE28 46890829 IC50 = 83 nM T92076 C45UEK 46890830 IC50 = 310 nM T92076 C9Q4RH 46890831 IC50 = 760 nM T92076 CPEG70 46891263 IC50 = 810 nM T92076 C5UI2F 46891264 IC50 > 30000 nM T92076 CQVA69 46891265 IC50 = 560 nM T92076 C6IMF2 46891266 IC50 = 220 nM T92076 CUCV79 46891319 IC50 = 2240 nM T92076 C6JZ8X 46891320 IC50 = 440 nM T92076 CSDV09 46891321 IC50 = 300 nM T92076 CO9Y6E 46891322 IC50 = 420 nM T92076 CE58QX 46891362 IC50 = 550 nM T92076 CZFT78 46891363 IC50 = 360 nM T92076 CHQ95U 46891364 IC50 = 92 nM T92076 CG2P6S 46891365 IC50 = 210 nM T92076 CME05N 46891415 IC50 = 150 nM T92076 C35OQN 46891416 IC50 = 200 nM T92076 CX5QY4 46891417 IC50 = 170 nM T92076 CMU51P 46891418 IC50 = 570 nM T92076 CU7G0V 46891464 IC50 = 74 nM T92076 CI2J5L 46891465 IC50 = 200 nM T92076 CER0U2 46891466 IC50 = 610 nM T92076 C6Y8LO 46891531 IC50 = 730 nM T92076 C5EI6L 46891532 IC50 = 140 nM T92076 CX3W6H 46891533 IC50 = 220 nM T92076 CCX0M5 46891590 IC50 = 140 nM T92076 CDS3Y4 46891591 IC50 = 540 nM T92076 C50DYX 46934584 EC50 = 17 nM T92076 C42EBH 46947061 EC50 = 10 nM T92076 CT3I7O 49864756 IC50 = 360 nM T92076 CMOS98 49864798 IC50 = 26 nM T92076 CN7AQ4 49864799 IC50 = 340 nM T92076 CANP45 49865336 IC50 = 2550 nM T92076 CB83YD 49865337 IC50 = 1950 nM T92076 CA0PK8 49865389 IC50 = 4690 nM T92076 C1CI4M 49865390 IC50 = 17000 nM T92076 C0OCF3 49865391 IC50 = 1900 nM T92076 C3Q8PC 49865392 IC50 = 2100 nM T92076 C2OZ4Q 49865393 IC50 = 1900 nM T92076 CKT41I 49865440 IC50 = 51 nM T92076 C9Y8HA 49865441 IC50 = 1820 nM T92076 C3R2OH 49865442 IC50 = 770 nM T92076 CZ3SB4 49865483 IC50 = 790 nM T92076 C5D8RF 49865484 IC50 > 10000 nM T92076 C84MFU 49865533 IC50 = 16 nM T92076 CBH83Y 49865681 IC50 = 2 nM T92076 C2VQ5N 49865952 EC50 = 350 nM T92076 C5Q8NZ 49866000 EC50 = 2700 nM T92076 CN5KG2 49866001 EC50 = 2200 nM T92076 C6YJV2 49866002 EC50 = 1400 nM T92076 CH6Q8M 49866003 EC50 = 870 nM T92076 CS78QB 49866004 EC50 = 620 nM T92076 CAYO91 49866054 EC50 = 280 nM T92076 CDHN69 49866112 EC50 = 58 nM T92076 C59OIM 49866113 EC50 = 3000 nM T92076 C24GNI 49866114 EC50 = 110 nM T92076 C2IO7B 51346981 IC50 = 4 nM T92076 CP62NF 51347014 IC50 = 5 nM T92076 C9ZK0F 52942726 EC50 = 251.19 nM T92076 C5WO8A 52942774 EC50 = 2511.89 nM T92076 C7VAT4 52944111 EC50 = 3981.07 nM T92076 CF1VH7 52945075 EC50 = 630.96 nM T92076 CSVB75 52945768 EC50 = 316.23 nM T92076 CX74IC 52946350 EC50 = 100 nM T92076 C6XNO0 52946369 EC50 = 31.62 nM T92076 C5Z8UV 52946370 EC50 = 100 nM T92076 CV41PS 52946552 IC50 > 10000 nM T92076 COZ12H 52947599 EC50 = 158.49 nM T92076 CADE86 52947600 EC50 = 79.43 nM T92076 C5LA1W 52948734 EC50 = 199.53 nM T92076 C6SRU2 52949984 EC50 = 398.11 nM T92076 C9I3NE 53317658 IC50 = 960 nM T92076 C4YFM8 53318971 IC50 = 11 nM T92076 CBD34V 53318993 IC50 = 18 nM T92076 CV3G9B 53321603 IC50 > 3000 nM T92076 C0GIP4 53324272 IC50 > 3000 nM T92076 CR89CV 53324273 IC50 = 2200 nM T92076 CL9I2S 53325542 IC50 > 3000 nM T92076 C0L6HP 53325543 IC50 = 23 nM T92076 CN6R1B 53326826 IC50 = 1500 nM T92076 CK86RJ 54582453 IC50 = 6 nM T92076 CSV2Y3 54583429 IC50 = 900 nM T92076 C0GBH6 54583478 IC50 = 350 nM T92076 C6XK4S 54583479 IC50 = 3500 nM T92076 CTS52H 54584449 IC50 = 18 nM T92076 CWO7B8 54585407 IC50 = 25 nM T92076 C58EQD 54586367 IC50 = 23 nM T92076 CU5IV1 54586368 IC50 = 50 nM T92076 CG8J7L 54587335 IC50 = 56 nM T92076 C1TUO0 54587336 IC50 = 3500 nM T92076 CH0WE1 54587337 IC50 = 300 nM T92076 C19UWQ 58938036 EC50 = 400 nM T92076 C4MN2U 58938040 EC50 = 60 nM T92076 C1G8ZC 58938049 EC50 = 286 nM T92076 CN7ZP6 58938052 EC50 = 1700 nM T92076 CFO62C 58938054 EC50 = 80 nM T92076 CX1AJ9 58938055 EC50 = 150 nM T92076 C4MW3Z 58938076 EC50 = 200 nM T92076 C04IPW 58938081 EC50 = 200 nM T92076 CY18FC 58938083 EC50 = 1000 nM T92076 CJK25L 58938087 EC50 = 450 nM T92076 CIUB04 58938101 EC50 = 150 nM T92076 C6X1LS 58938102 EC50 = 23 nM T92076 CL4RX7 58973485 EC50 = 158.49 nM T92076 C0FDV2 58973543 EC50 = 79.43 nM T92076 CBZ1Q4 59499324 EC50 = 90 nM T92076 C57OLB 59499339 EC50 = 300 nM T92076 CQKS81 59499356 EC50 = 80 nM T92076 CPZ6C9 59729011 EC50 = 4000 nM T92076 C31ASC 59729012 EC50 = 15000 nM T92076 CX4TA9 59729016 EC50 = 20000 nM T92076 CHQT92 59729027 EC50 = 3000 nM T92076 CVX9Z6 59729031 EC50 = 2000 nM T92076 CH35NC 59729041 EC50 = 4000 nM T92076 CAUR09 59729051 EC50 = 8000 nM T92076 CMSF35 59729055 EC50 = 15000 nM T92076 CRN80A 67404227 EC50 = 6000 nM T92076 COZ92N 67406778 EC50 = 190 nM T92076 CP0M3Q 67407227 EC50 = 290 nM T92076 CWK6J1 67410460 EC50 = 600 nM T92076 C49VFQ 69025930 EC50 = 1500 nM T92076 CQ6AS0 69026659 EC50 = 150 nM T92076 C0UGQ7 69028630 EC50 = 400 nM T92076 C6NVK9 69029375 EC50 = 100 nM T92076 CD8OC1 71579790 EC50 = 10000 nM T92076 C3VR8D 71579791 EC50 = 300 nM T92076 CQ7LC5 71579975 EC50 = 60 nM T92076 C3RY1P 71717737 EC50 = 600 nM T92076 C13PDJ 71719613 EC50 = 1000 nM T92076 CRD3Q6 72725152 EC50 = 300 nM T92076 CZ0K9V 72725153 EC50 = 1030 nM T92076 C8BIF7 72725211 EC50 = 175 nM T92076 CHI4F2 72725212 EC50 = 53 nM T92076 C7INA0 72725272 EC50 = 157 nM T92076 CTA63Q 72725273 EC50 = 18 nM T92076 CZ53XD 72725274 EC50 = 3 nM T92076 CQ8ZR4 72725275 EC50 = 2 nM T92076 CQ5Y7B 72725276 EC50 = 6 nM T92076 CAE7X0 72725335 EC50 = 17 nM T92076 CNM23Q 72725336 EC50 = 3 nM T92076 C1FUT4 72725337 EC50 = 4 nM T92076 CM2QZ6 72725338 EC50 = 19 nM T92076 C3HM6L 72725391 EC50 = 9 nM T92076 C7Z3EJ 72725392 EC50 = 9 nM T92076 C35FZS 72725393 EC50 = 20 nM T92076 C49BCG 72725441 EC50 = 10 nM T92076 C35VAF 73345828 EC50 = 200 nM T92076 CFQ4Z3 73347323 EC50 = 30 nM T92076 C6MAQ8 73348831 EC50 = 80 nM T92076 CH4BI3 73350366 EC50 = 200 nM T92076 C6VT0X 73350406 EC50 = 600 nM T92076 C9SBX8 73350407 EC50 = 30 nM T92076 C58IQN 73353384 EC50 = 80 nM T92076 CPNY69 73353385 EC50 = 30 nM T92076 C4C9LU 73353386 EC50 = 100 nM T92076 C5ZK6V 73353387 EC50 = 200 nM T92076 CFR05Y 73356416 EC50 = 1000 nM T92076 C8NVZ3 118163891 IC50 = 117.3 nM T92076 C84LHM 118173981 IC50 = 64.3 nM T92076 C42AZT 118181526 IC50 = 202.7 nM T92076 CR3KP8 122636590 IC50 = 17.7 nM T92076 C4T3QU 122636593 IC50 = 45.7 nM T92076 C4XDT0 122636607 IC50 = 457.1 nM T92076 C2WLF0 122636646 IC50 = 20 nM T92076 C8IS9G 122636658 IC50 = 58.7 nM T92076 C5N3RY 122636663 IC50 = 28.4 nM T92076 C6OU9D 122636665 IC50 = 21.8 nM T92076 CM4H7L 122636679 IC50 = 19.6 nM T92076 CJBC78 122636680 IC50 = 1332 nM T92076 C27NPS 122636684 IC50 = 27.6 nM T92076 C2QVH9 122636685 IC50 = 7.45 nM T92076 CMCZ89 122636699 IC50 = 50.8 nM T92076 CY6V7L 122636704 IC50 = 39.3 nM T92076 CZ3B1W 122636716 IC50 > 10000 nM T92076 CSAQ27 122636728 IC50 = 9.62 nM T92076 C2TYU1 122636753 IC50 = 21.6 nM T92076 CSVN38 122636757 IC50 = 489.1 nM T92076 CELN34 122636769 IC50 = 77.2 nM T92076 CQ0K8J 135401099 IC50 = 250 nM T92076 CX0JF2 135418418 IC50 = 300 nM T92076 CX7KB1 135422953 IC50 = 200 nM T92076 CU79GZ 135423282 IC50 = 140 nM T92076 C0ZG4P 135430131 IC50 = 95 nM T92076 CRIQ31 135430601 IC50 = 250 nM T92076 C9NDE1 135454814 IC50 = 100 nM T92076 CJS9A5 135457428 IC50 = 800 nM T92076 CPTX86 135464286 IC50 = 1600 nM T92076 C8E6VF 135464340 IC50 = 5.5 nM T92076 C3RWQ4 135483641 IC50 = 1600 nM T92076 C8KB6F 135492578 IC50 = 190 nM T92076 CN1SH4 135494510 IC50 = 1900 nM T92076 CKE1D2 135500059 IC50 = 300 nM T92076 CI51AJ 135507431 IC50 = 1100 nM T92076 CZDB71 135508434 IC50 = 120 nM T92076 CBS5N6 135517367 IC50 = 520 nM T92076 CV14PT 135524612 IC50 = 700 nM T92076 CX7Q1V 135537654 IC50 = 800 nM T92076 C5XYH1 135540474 IC50 = 170 nM T92076 CQ7Y0X 135543639 IC50 = 1600 nM T92076 C9YQ8Z 135543644 IC50 = 210 nM T92076 C53EHR 135795480 IC50 > 10000 nM T92076 CM2A9K 135903547 IC50 = 40 nM T92076 C2MPO5 135964370 IC50 = 200 nM T92076 C5LV7U 135964371 IC50 = 200 nM T92076 C1IR6C 135964374 IC50 = 140 nM T92076 C8ZGS6 135964376 IC50 = 160 nM T92076 C6EDB8 136030602 IC50 = 7.4 nM T92076 CJ08AR 136030614 IC50 = 3.5 nM T92076 C69MGK 136030615 IC50 = 4.1 nM T92076 CZ61NS 136030677 IC50 = 2900 nM T92076 C35JXR 136030692 IC50 = 1.7 nM T92076 CK4L2W 136030703 IC50 = 2.3 nM T92076 C3W4LU 136030746 IC50 = 12 nM T92076 C1FG6E 136030747 IC50 = 12 nM T92076 CZ98LU 136030753 IC50 = 2 nM T92076 CHZ64P 136030755 IC50 = 4.6 nM T92076 CT47ED 136032585 IC50 > 10000 nM T92076 CGEY37 136032586 IC50 > 10000 nM T92076 CSCD29 136032587 IC50 = 10 nM T92076 C0JXN6 136032594 IC50 > 10000 nM T92076 C06VFX 136032596 IC50 = 110 nM T92076 C7LE1T 136032598 IC50 = 320 nM T92076 CPR78N 136032621 IC50 = 76 nM T92076 C3TR5L 136032623 IC50 > 10000 nM T92076 CK65BJ 136032632 IC50 > 10000 nM T92076 CD2V9J 136032634 IC50 = 5300 nM T92076 CM3VD9 136045156 IC50 > 30000 nM T92076 C6Q9EW 136048766 IC50 = 600 nM T92076 C3ETP1 136059337 IC50 = 5.2 nM T92076 C3FZ1T 136059339 IC50 = 14 nM T92076 CC8H6J 136059340 IC50 = 7.6 nM T92076 CTZ3Q5 136059341 IC50 = 4.4 nM T92076 C0LA7G 136059342 IC50 = 23 nM T92076 CA0KY5 136059343 IC50 = 30 nM T92076 CQHP38 136059345 IC50 = 150 nM T92076 CH0VU4 136059346 IC50 = 3.4 nM T92076 CO34ST 136059347 IC50 = 17 nM T92076 CHJ98L 136059348 IC50 = 7.3 nM T92076 C4N7AI 136059349 IC50 = 6.6 nM T92076 C9ILF4 136059351 IC50 = 8.5 nM T92076 C6V2FP 136059356 IC50 = 25 nM T92076 C71GOL 136059370 IC50 = 2.3 nM T92076 CMTA04 136059372 IC50 = 31 nM T92076 C5S6OZ 136059376 IC50 = 31 nM T92076 C2NC5Z 136071244 IC50 = 31 nM T92076 CA6OC8 136071254 IC50 = 4.7 nM T92076 CO63TY 136071339 IC50 = 2.4 nM T92076 C3X8FC 136071531 IC50 = 320 nM T92076 C7GH3T 136072082 IC50 = 6.7 nM T92076 C9LZG5 136086811 IC50 = 97 nM T92076 C7LR0P 136110293 IC50 = 4.9 nM T92076 CUN01M 136141561 IC50 = 11 nM T92076 CQ3WH0 136141563 IC50 = 45 nM T92076 C34GPC 136141575 IC50 = 2.2 nM T92076 C60ZPK 136188834 IC50 = 380 nM T92076 CG6O8L 136188835 IC50 = 1.7 nM T92076 CSD8F7 136188836 IC50 = 3 nM T92076 C41UJN 136188837 IC50 = 4.2 nM T92076 CIK49P 136188838 IC50 = 4.8 nM T92076 CHW7P3 136188839 IC50 = 6 nM T92076 C2YF6M 136188840 IC50 = 6.1 nM T92076 C5AW8Z 136188841 IC50 = 11 nM T92076 C96DYG 136188842 IC50 = 11 nM T92076 CZ7S9J 136188843 IC50 = 13 nM T92076 CV1O7Y 136188844 IC50 = 81 nM T92076 C1HYA5 136199394 IC50 = 97 nM T92076 CEI91J 136199395 IC50 > 10000 nM T92076 C26GVI 136199396 IC50 > 10000 nM T92076 C5ME1N 136199397 IC50 = 400 nM T92076 CEB94Q 136199398 IC50 > 10000 nM T92076 CY16LP 136199399 IC50 = 700 nM T92076 CWP68O 137628638 EC50 = 50 nM T92076 CTYM47 137635178 EC50 = 12.59 nM T92076 C8JQN3 137637346 EC50 = 125.89 nM T92076 CZVA32 137638587 EC50 = 19.95 nM T92076 CQKN83 137638744 EC50 = 1584.89 nM T92076 C3O5PF 137638922 EC50 = 100 nM T92076 CG2T5Q 137641303 EC50 = 39.81 nM T92076 C2GKZ8 137644557 EC50 = 5.012 nM T92076 CB35FI 137645663 EC50 = 7.943 nM T92076 C7ZH2S 137646931 EC50 = 31.62 nM T92076 CB3C0F 137649972 EC50 = 3162.28 nM T92076 CC62LN 137652733 EC50 = 501.19 nM T92076 C9W2LX 137653796 EC50 = 39.81 nM T92076 CMUD47 137656029 EC50 = 39.81 nM T92076 CUA3H6 137658989 EC50 = 398.11 nM T92076 C7GCM5 137660522 EC50 = 7.943 nM T92076 CT4U9P 137661671 EC50 = 15.85 nM T92076 CZ83QK 145960490 EC50 = 93 nM T92076 C0G5BR 145960500 EC50 = 120 nM T92076 CC18GK 145960734 EC50 = 230 nM T92076 CA3XU2 145960800 EC50 = 430 nM T92076 CQGC21 145961658 EC50 = 600 nM T92076 C21JHZ 145962096 EC50 = 380 nM T92076 CNG8P5 145962145 EC50 = 8800 nM T92076 CQRC26 145962681 EC50 = 1100 nM T92076 CDQ0A1 145963186 EC50 = 50 nM T92076 C0PC7N 145963392 EC50 = 450 nM T92076 C4PCO6 145963561 EC50 = 320 nM T92076 CB9NF6 145963580 EC50 = 17 nM T92076 D02BCM 683379 IC50 = 3500 nM T92076 D04HDO 947434 IC50 = 14000 nM T92076 D04PHG 135515453 IC50 = 97 nM T92076 D0F4MI 135565722 IC50 = 0.94 nM T92076 D0HS5P 9882793 EC50 = 310 nM T92076 D0I1GV 44405854 IC50 = 270 nM T92076 D0Z8YZ 52943938 EC50 = 25.12 nM T64074 D0KV6C 53258905 IC50 = 0.069 nM T64074 CK4H5M 65087 IC50 = 142.58 nM T64074 C83GUS 213752 IC50 = 7.9 nM T64074 CZ17UA 11536300 IC50 = 1.01 nM T64074 C6K9EH 11573029 IC50 = 0.19 nM T64074 C1XJI4 11645134 IC50 = 0.02 nM T64074 CDFB07 11666585 IC50 = 0.29 nM T64074 CRUQ79 11673839 IC50 = 2.89 nM T64074 C19BQV 11688044 IC50 = 0.05 nM T64074 CE4G3V 23729147 IC50 = 0.03 nM T64074 CEK8R6 24777136 IC50 = 0.02 nM T64074 CBQ4V8 24978486 IC50 = 0.08 nM T64074 CWDC04 25003843 IC50 = 0.04 nM T64074 C2NC9B 25007428 IC50 = 0.11 nM T64074 C64DXG 44242661 IC50 = 0.32 nM T64074 CYV0D9 57576574 IC50 = 0.03 nM T64074 CLJ4S9 66924089 IC50 = 10.55 nM T64074 C4Y0HU 67301757 IC50 = 1.39 nM T64074 CM7E0A 132574708 IC50 = 0.11 nM T64074 CSCO64 136168051 IC50 = 1800 nM T64074 CG17QK 136168052 IC50 = 42200 nM T64074 CM10NY 137631470 IC50 = 1.77 nM T64074 C7N6WS 137636390 IC50 = 0.27 nM T64074 COE67T 137637328 IC50 = 0.25 nM T64074 CN37OR 137639798 IC50 = 2.3 nM T64074 CW27XK 137644048 IC50 = 16.2 nM T64074 CO0U6R 137646091 IC50 = 13.59 nM T64074 CIZQ40 137652049 IC50 > 10000 nM T64074 CJY3M0 137654933 IC50 = 334.3 nM T64074 CHK07O 137659411 IC50 > 10000 nM T64074 CWE0T6 137659579 IC50 = 12.31 nM T64074 C8ID1Y 145975543 IC50 = 244000 nM T64074 CC0J9B 146156039 IC50 < 0.02 nM T21653 D0K8KX 5280343 IC50 = 5090 nM T21653 D00UZR 5330286 IC50 > 5000 nM T21653 D0E3TC 44259 IC50 = 1.31 nM T21653 D0T3ME 156422 IC50 > 30000 nM T21653 C63WLY 89644 IC50 > 10 ug.mL-1 T21653 C5JE2Z 104860 IC50 = 2.2 ug.mL-1 T21653 CI1NA5 159926 IC50 > 10 ug.mL-1 T21653 CYBA43 177458 IC50 > 10 ug.mL-1 T21653 C8IAR2 5281657 IC50 = 33000 nM T21653 CI68PW 5283685 IC50 > 100000 nM T21653 CXK0S6 5283727 IC50 > 100000 nM T21653 CDQ3M7 5359485 IC50 = 0.95 ug.mL-1 T21653 C54BYP 5360741 IC50 = 4 ug.mL-1 T21653 C4G9WR 9547398 IC50 > 100000 nM T21653 C76CUP 9547698 IC50 > 100000 nM T21653 CR8DA1 10024683 IC50 > 100000 nM T21653 CLA93G 10047202 IC50 > 100000 nM T21653 C3LCH5 10047545 IC50 > 100000 nM T21653 C4CP7K 10423452 IC50 = 15600 nM T21653 C83QWV 10714343 IC50 = 29400 nM T21653 C8G5WP 11210533 IC50 = 3770 nM T21653 CL7X4Q 11530963 IC50 = 43000 nM T21653 CDGF78 15282555 IC50 = 1800 nM T21653 CW2XK6 16050925 IC50 = 840 nM T21653 C7YG1N 24759534 IC50 = 15 nM T21653 CCPS81 24764502 IC50 > 35000 nM T21653 CJH19T 24894883 IC50 = 4900 nM T21653 CJ14YB 24894884 IC50 = 2000 nM T21653 CHVU39 24894885 IC50 = 3600 nM T21653 CP7QT2 24894995 IC50 = 1800 nM T21653 CF4N9X 24895100 IC50 = 34000 nM T21653 CN13JF 24899915 IC50 = 0.75 ug.mL-1 T21653 CBWR97 24899916 IC50 = 0.35 ug.mL-1 T21653 C9F2JD 24899917 IC50 > 10 ug.mL-1 T21653 C64MTI 24900160 IC50 = 2.6 ug.mL-1 T21653 CO2I6Q 24900161 IC50 = 4 ug.mL-1 T21653 C4GI6J 25178540 IC50 = 9700 nM T21653 CJ5U1X 42639664 IC50 = 3.8 ug.mL-1 T21653 C8NA4L 53384644 IC50 > 30000 nM T21653 C9ZFS1 54764923 IC50 > 100000 nM T21653 C9DX3J 56649281 IC50 = 4.95 nM T21653 CXJ63M 59603829 IC50 = 19 nM T21653 CQEU96 59603842 IC50 = 4.2 nM T21653 CV63UL 67240318 IC50 > 10000 nM T21653 C5DGR9 69036886 IC50 = 5 nM T21653 C1V3NZ 73425588 IC50 = 7.97 nM T21653 C3UC9H 73891099 IC50 = 2510 nM T21653 CV8QX0 76310169 IC50 = 29800 nM T21653 CA5L4W 76324771 IC50 > 30000 nM T21653 C9GO0P 76328313 IC50 = 10000 nM T21653 C39FTZ 76335685 IC50 > 100000 nM T21653 C1HW4B 89735655 IC50 = 200 nM T21653 CL0YO5 118443595 IC50 > 100 nM T21653 C3KLI5 118723185 IC50 > 100000 nM T21653 CQCX41 118737057 IC50 > 10000 nM T21653 CBSW14 129116690 IC50 = 400 nM T21653 CPHG43 135567142 IC50 = 2 nM T21653 COG2M5 136242661 Ki = 1.7 nM T21653 C04YDK 137248544 Ki = 11 nM T21653 CMB78I 137301774 Ki = 8.6 nM T21653 C2MD1Q 155513187 IC50 > 10000 nM T21653 D00ERW 44444843 Ki > 1503 nM T21653 D06QWO 14824655 IC50 > 10 ug.mL-1 T21653 D09PTP 57325421 IC50 = 26 nM T21653 D0A1CM 5281855 IC50 = 510 nM T21653 D0G3SZ 6918469 IC50 = 6.6 ug.mL-1 T21653 D0X1RH 16051023 IC50 = 2000 nM T17986 CTG1H0 53492732 IC50 = 60 nM T17986 C4Z1RG 67465326 IC50 > 5000 nM T17986 C78LNX 118572065 Ki = 70 nM T17986 CKN23I 134133285 IC50 = 1980 nM T17986 CXI6A2 134134567 IC50 = 1350 nM T17986 CCRF30 134134857 IC50 = 2710 nM T17986 C19OZF 134135375 IC50 = 7750 nM T17986 C54HDM 134135389 IC50 = 1870 nM T17986 CTE31R 134137113 IC50 = 3340 nM T17986 CO52FX 134137743 IC50 = 4440 nM T17986 CJ0L2E 134139550 IC50 = 2650 nM T17986 CT2J1B 134142243 IC50 = 1560 nM T17986 C2Y3KW 139211326 IC50 > 2500 nM T17986 CAJ94H 155538504 IC50 > 5000 nM T17986 C75ENB 155538833 IC50 > 5000 nM T17986 CPY0B1 155540279 IC50 > 5000 nM T17986 CQ8EU9 155540351 IC50 > 5000 nM T17986 C3SLV6 155541578 IC50 > 5000 nM T17986 CJ3SF0 155542049 IC50 > 5000 nM T17986 CYPH45 155542586 IC50 > 2500 nM T17986 CF3IE0 155542683 IC50 = 315 nM T17986 C9TWY6 155542713 IC50 > 2500 nM T17986 C1P6ZK 155542893 IC50 > 5000 nM T17986 C7V0NB 155544716 IC50 > 5000 nM T17986 C8I2CL 155545225 IC50 = 394 nM T17986 CWB86N 155546955 IC50 > 1250 nM T17986 C2OHG1 155546957 IC50 > 2500 nM T17986 C2DY0H 155547180 IC50 > 2500 nM T17986 CFJK12 155547766 IC50 > 2500 nM T17986 CXVM95 155547840 IC50 > 1250 nM T17986 C3GZP6 155547915 IC50 > 1250 nM T17986 CY2RI3 155548857 IC50 > 5000 nM T17986 CBW5H1 155548936 IC50 > 2500 nM T17986 CTG91O 155549667 IC50 = 127 nM T17986 C5W6GC 155550181 IC50 > 2500 nM T17986 CBA42L 155550828 IC50 > 10000 nM T17986 COAX09 155550957 IC50 > 5000 nM T17986 CM0N8B 155550993 IC50 > 10000 nM T17986 CH50KG 155551023 IC50 = 681 nM T17986 C8TZ2H 155552001 IC50 > 10000 nM T17986 CA95GN 155552788 IC50 = 810 nM T17986 CF8H7X 155553332 IC50 = 126 nM T17986 CWE04H 155554866 IC50 = 211 nM T17986 CE6NL4 155555991 IC50 > 2500 nM T17986 CN6WA2 155556614 IC50 = 160 nM T17986 C5SBY9 155557240 IC50 = 88 nM T17986 C5C6GK 155557835 IC50 = 108 nM T17986 C8N2FZ 155557917 IC50 = 320 nM T17986 CHR6N8 155558797 IC50 > 2500 nM T17986 C74JAU 155559342 IC50 > 10000 nM T17986 C1XA8H 155560365 IC50 = 86 nM T17986 CJO5K6 155560444 IC50 > 2500 nM T17986 CWK90R 155560721 IC50 = 613 nM T17986 C8IX9W 155560875 IC50 > 1250 nM T17986 C8K0IE 155561239 IC50 > 10000 nM T17986 COT94K 155563932 IC50 = 880 nM T17986 CPA5R9 155564424 IC50 > 5000 nM T17986 C2CAX7 155564971 IC50 > 2500 nM T17986 C18OAD 155567358 IC50 > 5000 nM T17986 CKXG20 155568357 IC50 > 10000 nM T17986 CEIC47 155568678 IC50 > 10000 nM T17986 CW52CQ 155568924 IC50 = 773 nM T17986 CJI41G 155569031 IC50 > 10000 nM T17986 D09CLP 439155 IC50 = 6400 nM T23787 D03BNU 59604787 IC50 > 10000 nM T23787 CFAB91 96506 Ki = 1290 nM T23787 CZ8NC9 733090 IC50 > 1000000 nM T23787 CV32NS 3431969 IC50 = 7400 nM T23787 C94AZF 5720233 IC50 = 22900 nM T23787 C2CZ1O 7087401 IC50 = 490 nM T23787 CT0U8L 9815029 IC50 > 100000 nM T23787 C2P9NE 9858287 IC50 = 2320 nM T23787 CQH51Y 53374134 IC50 > 1000000 nM T23787 C60IAQ 58619539 IC50 = 575 nM T23787 CBC0Y3 73669296 IC50 = 2600 nM T23787 C8IQW5 76310213 IC50 = 55000 nM T23787 C64ZIP 76310214 IC50 > 500000 nM T23787 CHLA09 76313903 IC50 = 11000 nM T23787 C6LDE1 76313904 IC50 = 26000 nM T23787 C4RKN2 76317433 IC50 = 9100 nM T23787 C0LE8B 76317434 IC50 = 8700 nM T23787 CQ63TU 76317435 IC50 > 1000000 nM T23787 C0COF3 76321167 IC50 = 7000 nM T23787 CU2RY9 76321168 IC50 > 500000 nM T23787 CS7H9O 76328353 IC50 = 3400 nM T23787 CMAJ92 76328354 IC50 > 500000 nM T23787 C3NHU8 76328355 IC50 > 1000000 nM T23787 C8INV7 76328356 IC50 = 13000 nM T23787 C31DEP 76328357 IC50 > 1000000 nM T23787 CG31TZ 76332025 IC50 = 9600 nM T23787 CS0GP8 76332026 IC50 > 1000000 nM T23787 CD9Y0S 76335629 IC50 = 8400 nM T23787 CCF41B 76335630 IC50 > 10000000 nM T23787 CQSU96 91668553 IC50 = 104 nM T23787 CGDW51 91668554 IC50 = 11 nM T23787 C1BX7Z 91668556 IC50 = 2010 nM T23787 C9LM8K 91668557 IC50 = 21 nM T23787 CF0MU1 118735141 IC50 = 1570 nM T23787 CPR4H8 118735142 IC50 = 13700 nM T23787 C1F8YJ 118735143 IC50 = 111 nM T23787 C7V3SG 118735144 IC50 = 24700 nM T23787 CU07TA 118735145 IC50 = 199 nM T23787 CS1WQ8 118735769 IC50 = 23 nM T23787 CFC42D 118735770 IC50 = 514 nM T23787 CMHZ30 118735771 IC50 = 815 nM T23787 CSB1V0 118735772 IC50 > 100000 nM T23787 CXN4E3 118735773 IC50 = 16400 nM T23787 C3OYE2 118735774 IC50 = 343 nM T23787 C5U6TN 118735775 IC50 = 562 nM T23787 CB1TD9 118735776 IC50 = 830 nM T23787 C8TM3X 118735777 IC50 = 9830 nM T23787 CES82L 118735778 IC50 = 112 nM T23787 CJDN52 118735779 IC50 = 70900 nM T23787 C7WM8V 118735780 IC50 = 23100 nM T23787 C93NLH 118735781 IC50 = 86 nM T23787 CBAN54 118735782 IC50 = 2200 nM T23787 C78XED 118735783 IC50 = 531 nM T23787 CZOI63 118735784 IC50 = 14000 nM T23787 CF5RS3 118735785 IC50 = 256 nM T23787 CQTH95 118735786 IC50 = 633 nM T23787 CO46US 118735787 IC50 = 27 nM T23787 CEA1Q3 118735788 IC50 = 140 nM T23787 CQ3ZF9 118735789 IC50 = 20 nM T23787 CUS6C9 118735790 IC50 = 4 nM T23787 CPF65J 118735791 IC50 = 3 nM T23787 CK4XS8 118735793 IC50 = 114 nM T23787 CA6Q1T 122689236 IC50 = 3500 nM T23787 CBW5A7 122689285 IC50 = 49 nM T23787 CPZ8F9 122690573 IC50 = 38 nM T23787 CMI96Q 122690579 IC50 = 26 nM T23787 CEY07L 122690584 IC50 = 116 nM T23787 CNL3D8 122690595 IC50 = 11 nM T23787 CIT04P 122690602 IC50 = 35 nM T23787 CWB07X 122690613 IC50 = 31260 nM T23787 CV2ET1 122690615 IC50 = 265 nM T23787 C8U0VJ 122690619 IC50 = 59 nM T23787 C2PSJ3 122690641 IC50 = 1692 nM T23787 CY3M9U 122690654 IC50 = 73 nM T23787 CAC31L 122690672 IC50 = 74 nM T23787 CSO0W8 122690681 IC50 = 22 nM T23787 C97SNC 122690695 IC50 = 105 nM T23787 CSAV23 122690696 IC50 = 93 nM T23787 CAM94G 122690699 IC50 = 7020 nM T23787 C1N4MA 122690707 IC50 = 30 nM T23787 C6S9BW 122690708 IC50 = 56450 nM T23787 C8GRF1 122690737 IC50 = 106 nM T23787 C87KBS 122690767 IC50 = 38 nM T23787 CK74UB 122690768 IC50 = 4640 nM T23787 CN5FU9 122690771 IC50 = 9 nM T23787 C5VP3U 122690775 IC50 = 41 nM T23787 CHXA05 122690782 IC50 = 176 nM T23787 CPR80N 122690857 IC50 = 26500 nM T23787 CD50EH 122690862 IC50 = 3160 nM T23787 CK7X2C 122690886 IC50 = 62 nM T23787 C31OZR 122690891 IC50 = 15 nM T23787 C30YDX 122690933 IC50 = 4 nM T23787 CX4BZ9 122690935 IC50 = 2 nM T23787 C9JX8Z 122690977 IC50 = 17 nM T23787 CY8RI3 122690986 IC50 = 137 nM T23787 CH1U6B 122691005 IC50 = 33 nM T23787 CR79QC 122697986 IC50 = 104 nM T23787 CV1US4 122698052 IC50 = 499 nM T23787 CTRJ81 122698090 IC50 = 2640 nM T23787 CX29CB 122698115 IC50 = 85 nM T23787 CJV1R8 134463139 IC50 = 94 nM T23787 CBP5S0 134463146 IC50 = 159 nM T23787 D09FDZ 5466139 IC50 = 670 nM T23787 D0A8AL 25142799 IC50 = 207 nM T86271 D0K9IF 71666749 IC50 > 30000 nM T86271 CV4Q5S 704452 IC50 = 11 nM T86271 CDK30S 772885 IC50 = 123 nM T86271 C67LUP 24857841 IC50 = 2600 nM T86271 C6CZ1L 25110719 IC50 = 530 nM T86271 CJ2AK1 44589880 IC50 = 1100 nM T86271 CWC04O 57390845 Ki = 397 nM T86271 C4C3RA 57396284 Ki = 593 nM T86271 C0U3HP 57401348 Ki = 90 nM T86271 CL5MG9 57403100 Ki = 878 nM T86271 CN0P9L 57403256 Ki = 194 nM T55005 D0E3TC 44259 IC50 = 1.67 nM T55005 CV63UL 67240318 IC50 > 10000 nM T55005 C2MD1Q 155513187 IC50 > 10000 nM T20709 D01AZG 5073 Ki > 1000 nM T20709 D01ZII 2726 Ki = 158.49 nM T20709 D08CTT 21855 Ki = 407.38 nM T20709 D0B4TN 2381 Ki = 32.1 nM T20709 D0BZ7W 443879 Ki = 3.1 nM T20709 D0H3HM 60795 Ki > 1000 nM T20709 D0H7KF 5002 Ki = 125.89 nM T20709 D0L4YD 154059 Ki = 128.82 nM T20709 D0M0AM 11693 IC50 = 0.1585 nM T20709 D0M6VK 71183 Ki = 0.1413 nM T20709 D0Q9HF 187 EC50 = 10 nM T20709 D0RG3O 174174 Ki = 0.34 nM T20709 D0T0LM 4848 Ki = 13.8 nM T20709 D0T6QX 5736 Ki = 550 nM T20709 D0U7BW 5831 Ki = 24 nM T20709 D0V4QS 135398745 Ki = 12.59 nM T20709 D0VP1V 11434515 IC50 = 0.1995 nM T20709 D0Y5AM 444031 Ki = 8.6 nM T20709 D0Z1RV 135398737 Ki = 12.59 nM T20709 D07EFM 2230 Ki = 26 nM T20709 D0FD6D 11751922 Ki = 2900 nM T20709 D0I5XU 16065403 Ki = 0.115 nM T20709 D0K4HW 135409468 Ki = 290 nM T20709 D0N1HW 5311200 Ki > 10000 nM T20709 D02JNY 10030021 Ki = 50.12 nM T20709 D06ACX 6436265 Ki = 8.71 nM T20709 D06DZI 107780 Ki > 10000 nM T20709 D08YVT 9894173 Ki = 61 nM T20709 D09FYQ 9577995 EC50 = 5.7 nM T20709 D0A2OW 107867 Ki = 407 nM T20709 D0J8UV 9928284 IC50 > 10000 nM T20709 D0R1VL 132712 Ki = 173.78 nM T20709 D0VZ3D 129989 Ki = 6.457 nM T20709 C01PRU 1993 Ki = 1600 nM T20709 C45PUM 2551 EC50 = 154.88 nM T20709 C4AWJ9 2684 Ki = 1023.29 nM T20709 CKD46H 4022 Ki = 9120.11 nM T20709 C7VMZ3 4108 Ki = 38 nM T20709 C5H9CN 9287 Ki > 10000 nM T20709 C89UZB 18493 Ki = 13.2 nM T20709 CNZD18 36381 Ki = 1415 nM T20709 CRCD50 60809 EC50 = 6 nM T20709 C8E9XD 66007 IC50 = 6.7 nM T20709 CT0GD8 66266 Ki = 912.01 nM T20709 C3WKC6 68835 IC50 > 100000 nM T20709 C3S8RF 71792 EC50 = 844 nM T20709 CA3W0P 100826 IC50 > 100000 nM T20709 CBH8L0 156308 Ki = 2000 nM T20709 CVWA68 197841 Ki = 1690 nM T20709 C9XWA6 198914 Ki > 30000 nM T20709 CP2DY7 198967 Ki > 300000 nM T20709 CHLK79 214124 Ki = 18.5 nM T20709 CD65GI 315401 Ki = 7.23 nM T20709 C6OQ8S 410345 Ki = 9.48 nM T20709 CD8Z9H 424430 Ki = 35000 nM T20709 CX75UZ 598754 Ki > 19952.62 nM T20709 CC56KR 639794 Ki = 14791.08 nM T20709 C91GCI 657308 Ki = 0.382 nM T20709 CEGR96 657346 Ki = 8912.51 nM T20709 C24ERV 672747 EC50 = 371.54 nM T20709 C0NQC6 682264 EC50 = 120 nM T20709 CXC0Q5 683024 EC50 = 891 nM T20709 CSJ39D 698706 EC50 = 478.63 nM T20709 C4HCK5 729510 IC50 > 30000 nM T20709 C08WCU 851833 Ki > 19952.62 nM T20709 C3C2KZ 885513 EC50 = 354.81 nM T20709 CUD48J 952858 IC50 > 10000 nM T20709 C7OCV4 1045715 EC50 > 10000 nM T20709 CH5WR4 1421986 IC50 = 3700 nM T20709 C6YLU1 1505736 EC50 = 223.87 nM T20709 C4PMT9 1505737 EC50 = 154.88 nM T20709 CD83WM 1506223 EC50 = 177.83 nM T20709 C5NK4G 2091326 EC50 > 10000 nM T20709 CO84FN 2150723 EC50 > 10000 nM T20709 CW9SD2 2150737 EC50 > 10000 nM T20709 CUIZ43 2150760 EC50 > 10000 nM T20709 CPL49A 2157678 EC50 > 30000 nM T20709 CM64LI 2159295 EC50 = 1348.96 nM T20709 CS8N5X 2736067 Ki = 31622.78 nM T20709 CJ6D8N 3342390 Ki < 1000 nM T20709 CX8W7I 3377940 Ki > 300000 nM T20709 C37EXL 3480822 EC50 > 10000 nM T20709 CI7DF6 3675988 Ki = 87096.36 nM T20709 CX3S8T 4715419 Ki = 51286.14 nM T20709 C12BJA 4995951 Ki = 6.457 nM T20709 CS71UA 5189681 IC50 > 30000 nM T20709 C1JP8T 5204148 EC50 = 1819.7 nM T20709 CR5LG3 5310989 IC50 = 333.5 nM T20709 C3A1FO 6604789 Ki = 25118.86 nM T20709 CFN7L4 6604866 Ki = 295.12 nM T20709 C2IP0Y 7022778 Ki = 102329.3 nM T20709 CVSC58 7047822 Ki = 89125.09 nM T20709 C32TSZ 7141654 Ki = 208929.61 nM T20709 C7NJZ2 7141656 Ki = 29512.09 nM T20709 C7MBO3 9809330 Ki = 1.995 nM T20709 C80IET 9843967 Ki = 590 nM T20709 C1N0KW 9867847 Ki = 0.33 nM T20709 CQ4LC2 9872676 Ki = 3680 nM T20709 CDLB96 9889149 IC50 > 1000 nM T20709 CJ5K1D 9889312 Ki = 14.8 nM T20709 CUN81Q 9905249 Ki > 10000 nM T20709 C2U5LK 9905467 IC50 = 142.7 nM T20709 CYWQ50 9906447 Ki = 351 nM T20709 CDB9E1 9909907 Ki = 31.62 nM T20709 CXAV92 9911615 Ki = 1.995 nM T20709 CXAY37 9913341 Ki = 2.512 nM T20709 CRV17M 9931930 Ki = 1.995 nM T20709 C50NSR 9936450 Ki = 0.7762 nM T20709 CA2HR0 9937709 EC50 = 1.4 nM T20709 CQ04ZS 9950396 Ki = 300 nM T20709 C58KXV 9958728 EC50 = 1100 nM T20709 CYNT43 9968046 Ki = 616.6 nM T20709 CCM72P 9974222 IC50 = 69.7 nM T20709 C9FR0C 9998508 Ki = 1230.27 nM T20709 CV7R9F 10020040 Ki > 10000 nM T20709 CQZ0K4 10027177 EC50 > 50000 nM T20709 C2EUY0 10035109 Ki > 10000 nM T20709 C7I6DA 10035281 Ki = 900 nM T20709 CBJ63D 10043954 Ki = 1698.24 nM T20709 C2JZL1 10048222 IC50 > 1000 nM T20709 C9OQ2S 10066369 Ki = 741.31 nM T20709 CI6SD7 10066972 Ki = 1819.7 nM T20709 CCO72H 10082470 IC50 = 1200 nM T20709 C8NQ3I 10092649 Ki = 130 nM T20709 CG0O9Z 10109893 Ki = 794.33 nM T20709 CUT05R 10114698 Ki = 10.96 nM T20709 C90FZG 10139614 Ki = 14.13 nM T20709 C0PO3J 10142923 Ki = 2.512 nM T20709 CG78WP 10160073 Ki = 1 nM T20709 CZ8E9X 10160219 Ki = 1 nM T20709 C4TR5Q 10180872 Ki = 2.2 nM T20709 COR14Y 10203251 Ki = 1.995 nM T20709 CB69ND 10204457 Ki = 18.6 nM T20709 CJ5V2S 10225340 Ki = 9.05 nM T20709 C04QCB 10225881 Ki = 3.02 nM T20709 C6A5KD 10226456 Ki = 79.43 nM T20709 CO64WJ 10236758 IC50 = 177.83 nM T20709 C3W2YB 10248541 IC50 = 910 nM T20709 C3QGA5 10251795 EC50 > 50000 nM T20709 CW90FO 10261985 EC50 = 30 nM T20709 C1FCP7 10262466 Ki = 222 nM T20709 CH31DX 10267394 Ki > 10000 nM T20709 CC6RP7 10267601 IC50 = 62 nM T20709 CY3E5J 10274019 Ki = 0.07 nM T20709 CU89JD 10314060 Ki > 10000 nM T20709 CD1C0H 10315426 Ki = 891.25 nM T20709 C6S7GK 10354348 IC50 > 100000 nM T20709 C7BZ1R 10358345 IC50 = 367 nM T20709 CBSA40 10360219 Ki = 173.78 nM T20709 C69KIB 10385855 IC50 > 10000 nM T20709 CL7D2U 10421982 Ki = 410 nM T20709 C5BEJ0 10442081 EC50 = 240 nM T20709 CIRS06 10442337 EC50 = 67 nM T20709 CEF2O6 10478367 Ki > 10000 nM T20709 C1GT3O 10487582 IC50 = 800 nM T20709 C8COH6 10499832 IC50 = 2388.2 nM T20709 CS1P4M 10511551 IC50 = 975 nM T20709 CP9M5J 10516408 IC50 = 3788.8 nM T20709 C37PDA 10518821 IC50 = 31125.4 nM T20709 C6T1JW 10521205 IC50 = 836.1 nM T20709 C4WZ3R 10522202 IC50 = 1167.2 nM T20709 C5MB2F 10522336 IC50 = 1577.9 nM T20709 C0K9HN 10538337 IC50 = 13042.1 nM T20709 C3Y6JB 10546275 IC50 = 282.3 nM T20709 CI3GQ6 10547222 IC50 = 2123.9 nM T20709 C6XKZ9 10549581 IC50 = 4162.1 nM T20709 CFD40Z 10567192 IC50 = 108.7 nM T20709 C4AL8Q 10569816 IC50 = 1756.1 nM T20709 CB37SH 10573693 IC50 = 7708.4 nM T20709 C71VMD 10591874 IC50 = 472.8 nM T20709 C94VUE 10592484 IC50 = 2196.7 nM T20709 C51LBK 10593954 IC50 = 1132.1 nM T20709 CH2QU8 10594386 IC50 = 19581.2 nM T20709 CY54RA 10595006 Ki = 1730 nM T20709 CZRJ60 10610375 IC50 = 13691.8 nM T20709 CX01SE 10611310 IC50 = 3226.4 nM T20709 CO3H7D 10614695 IC50 = 8428.6 nM T20709 CJL4R1 10636001 IC50 = 1409.3 nM T20709 C09XHV 10638050 IC50 = 701 nM T20709 C5VWL8 10641009 IC50 = 134.7 nM T20709 CONH15 10663572 IC50 = 146.3 nM T20709 C6WQ2Z 10664532 IC50 = 1740.6 nM T20709 C8CF4H 10666533 IC50 = 2224.5 nM T20709 C0AV8X 10678449 IC50 = 1100 nM T20709 C32KQX 10684720 IC50 = 524 nM T20709 C32EGP 10686988 IC50 = 572.7 nM T20709 C9O6LN 10688349 IC50 = 8122.8 nM T20709 CEB3A5 10726038 IC50 = 495 nM T20709 CC21XD 10755732 IC50 = 656.3 nM T20709 CHL29Z 10755733 IC50 = 742.6 nM T20709 C4JXA3 10757736 IC50 = 4246.3 nM T20709 CPQ7Z3 10760249 IC50 = 138 nM T20709 C5P3DQ 10761219 IC50 = 7422 nM T20709 CX4LT3 10777692 IC50 = 10383 nM T20709 CA4QI2 10782321 IC50 = 63337.5 nM T20709 C4N9IT 10782462 IC50 = 167.6 nM T20709 C6FC0M 10784004 IC50 = 1160.8 nM T20709 CV8TE0 10785471 IC50 = 566.2 nM T20709 CW5TJ6 10797864 IC50 = 49 nM T20709 C9SEA6 10806268 IC50 = 617.1 nM T20709 CGR64V 10808719 IC50 = 2775.5 nM T20709 CK1D3J 10827157 IC50 = 896.9 nM T20709 CR1X5L 10829928 IC50 = 8392.3 nM T20709 CB7E2O 10846833 IC50 = 14500 nM T20709 CH9WK6 10851853 IC50 = 432.4 nM T20709 CX6AP3 10852843 IC50 = 7900 nM T20709 C5PRT6 10854879 IC50 = 1250 nM T20709 C8HI5L 10854880 IC50 = 258.8 nM T20709 CZ85AJ 10862395 Ki = 3.981 nM T20709 CHE9P4 10865439 Ki = 16.6 nM T20709 CCM3L9 10870954 Ki = 26915.35 nM T20709 C2YNC5 10871551 Ki = 831.76 nM T20709 CFAD04 10874119 Ki = 72.44 nM T20709 CTV95B 10880435 Ki = 2398.83 nM T20709 CFP75Y 10907744 EC50 > 100000 nM T20709 C4A8QE 10916286 Ki = 1949.84 nM T20709 CQLR32 10919522 Ki = 2.3 nM T20709 CC12TE 10925451 Ki = 741.31 nM T20709 C5LVY0 10949838 Ki = 3.02 nM T20709 CE05FM 10951142 Ki = 97.72 nM T20709 C1WF5L 10952349 EC50 = 0.6 nM T20709 CA6X3W 10952416 EC50 = 4.7 nM T20709 C3K6JV 10957754 Ki = 1698.24 nM T20709 CN4QT5 10963509 Ki = 15.3 nM T20709 C4WV8L 10969390 Ki = 436.52 nM T20709 CTYZ13 10969696 Ki = 4168.69 nM T20709 C41PXY 10982070 Ki = 190.55 nM T20709 C9E2MP 10984804 Ki > 1700 nM T20709 C2W3GM 11000399 Ki = 8317.64 nM T20709 C6NH9T 11001809 Ki = 13182.57 nM T20709 CQ8D4K 11004046 Ki = 15.14 nM T20709 C6BG1N 11006792 Ki = 43 nM T20709 CU4Z0J 11011332 Ki = 7413.1 nM T20709 CZK86F 11011757 Ki = 371.54 nM T20709 CVA6U9 11012653 Ki = 1000 nM T20709 CPM1Z7 11012712 Ki = 4168.69 nM T20709 CW23BJ 11013666 Ki = 128.82 nM T20709 C6TF5I 11015312 Ki = 67.61 nM T20709 CBA37I 11017197 EC50 > 100000 nM T20709 C7Y1DO 11024241 Ki = 1995.26 nM T20709 C3L9ON 11034265 Ki = 645.65 nM T20709 CHDT49 11039424 Ki = 14 nM T20709 CP9OJ6 11045444 Ki = 616.6 nM T20709 C4ZUH9 11048067 Ki = 109.65 nM T20709 CQ8O3Y 11057942 Ki > 12302.69 nM T20709 CIG31V 11061341 Ki = 11 nM T20709 CT3XN5 11071537 Ki = 19.95 nM T20709 CO3C6Q 11072401 EC50 = 1 nM T20709 C5VQ6H 11079969 Ki = 15.14 nM T20709 C1TFO4 11081520 EC50 = 3900 nM T20709 CWS56C 11092603 Ki = 72.44 nM T20709 C02MPO 11099206 Ki = 1230.27 nM T20709 CSNA03 11101362 Ki = 363.08 nM T20709 CF81CB 11110049 Ki = 87096.36 nM T20709 C7ROJ1 11112362 Ki = 1348.96 nM T20709 C9CY0M 11120347 Ki = 1412.54 nM T20709 C2C4AN 11131099 Ki = 8511.38 nM T20709 CB37ZA 11135606 EC50 > 100000 nM T20709 C1T9WI 11143997 Ki = 7.079 nM T20709 C9FNM4 11431811 Ki = 0.0078 nM T20709 CGCF61 11515738 Ki < 100000 nM T20709 CY63VP 11523050 Ki = 46773.51 nM T20709 C07AJD 11530306 Ki < 100000 nM T20709 CWUP85 11542982 Ki < 100000 nM T20709 C6D1MA 11584660 IC50 = 158.49 nM T20709 CEHP14 11586481 Ki < 100000 nM T20709 CP3Y7J 11588240 Ki < 100000 nM T20709 CQ5PI4 11622544 Ki < 100000 nM T20709 CF2ZC0 11651360 Ki < 100000 nM T20709 CHKN81 11653111 Ki < 100000 nM T20709 C27XOS 11660220 Ki < 100000 nM T20709 C0N4BQ 11672895 Ki < 100000 nM T20709 CN4Z5C 11679149 IC50 > 10000 nM T20709 CW8CE2 11694118 Ki < 100000 nM T20709 CF8MO2 11694119 Ki < 100000 nM T20709 C9BF1S 11715398 Ki < 100000 nM T20709 CEY7J3 11729182 Ki = 9772.37 nM T20709 CPG15O 11743399 IC50 > 1000 nM T20709 C4QVR6 11748799 Ki = 81.28 nM T20709 CQLP36 11759058 Ki = 46773.51 nM T20709 CW3GA7 11759212 Ki = 331.13 nM T20709 CBM05D 11759379 Ki = 1905.46 nM T20709 CFZ4L5 11767229 Ki = 30 nM T20709 C9LUA7 11773414 Ki = 300 nM T20709 C39HRB 11793999 IC50 = 951.2 nM T20709 CT4F2C 11808040 Ki = 97.72 nM T20709 CXQ10I 11808946 Ki = 660.69 nM T20709 C6EXD3 11808947 Ki = 602.56 nM T20709 C30WRH 11809446 Ki = 14791.08 nM T20709 CJIA51 11828362 Ki = 31 nM T20709 CR9FJ2 11833737 Ki = 3235.94 nM T20709 CZ3AX9 11834199 Ki = 457.09 nM T20709 C8JQL7 11957735 IC50 > 10000 nM T20709 CL91TM 11968014 IC50 = 3.802 nM T20709 CYU4P5 12739458 Ki = 1784 nM T20709 CJF73M 12872436 Ki = 11.22 nM T20709 CR10FQ 13567080 Ki = 6.166 nM T20709 CS54WY 14537188 Ki = 566 nM T20709 CA87RQ 14660293 IC50 = 100000 nM T20709 CMO81H 14925759 EC50 = 588.84 nM T20709 CZ16XJ 15157137 Ki = 1.5 nM T20709 C5VC9Z 15157138 Ki = 4.6 nM T20709 C7VT5X 15157139 Ki = 65.6 nM T20709 CD3MI7 15157140 Ki = 209 nM T20709 CY80DC 15157141 Ki = 173 nM T20709 CUB5X2 16038385 EC50 = 199.53 nM T20709 CZ47FJ 16071018 EC50 = 251.19 nM T20709 C3T0UX 16085999 Ki = 29 nM T20709 CWI32N 16086000 Ki = 41 nM T20709 C71HBL 16086001 Ki = 20 nM T20709 C7EM1G 16086003 Ki = 480 nM T20709 CFU72Z 16086004 Ki = 290 nM T20709 CTOM27 16086005 Ki = 24 nM T20709 C7WF9Y 16086059 Ki = 42 nM T20709 C05YVJ 16086060 Ki = 39 nM T20709 CMQ8U3 16086061 Ki = 92 nM T20709 CEI8G1 16086062 Ki = 31 nM T20709 CGB89M 16086063 Ki = 11 nM T20709 CUS73E 16086064 Ki = 48 nM T20709 CHJ07L 16086065 Ki = 150 nM T20709 CEV68D 16086066 Ki = 53 nM T20709 CIX9M7 16086067 Ki = 120 nM T20709 C1XZ7V 16094783 Ki = 63.1 nM T20709 CO16DS 16094788 Ki = 12.59 nM T20709 CYN71L 16094791 Ki = 79.43 nM T20709 C2HK7W 16094793 Ki = 158.49 nM T20709 C9R0JN 16094810 Ki = 158.49 nM T20709 CTYI57 16115796 Ki = 1.995 nM T20709 C5HSD9 16115797 Ki = 1 nM T20709 CQ85FK 16115798 Ki = 1.202 nM T20709 CR1Z4N 16115799 Ki = 1.259 nM T20709 CLA6E0 16115800 Ki = 3.467 nM T20709 CTE0R7 16115942 Ki = 1.82 nM T20709 C7IC9E 16115944 Ki = 0.871 nM T20709 CQ3C9X 16115946 Ki = 0.7079 nM T20709 C0JGY1 16115950 Ki = 3.311 nM T20709 CZ67DO 16115951 Ki = 2.344 nM T20709 CO3YU4 16116082 Ki = 0.4677 nM T20709 C3IKJ0 16116084 Ki = 0.871 nM T20709 CWU6P3 16123945 EC50 = 630.96 nM T20709 CQ3HO2 16309462 EC50 = 410 nM T20709 C1G3IE 16371349 EC50 = 2300 nM T20709 CZ2IS9 16660294 Ki > 10000 nM T20709 C50JQV 17413870 EC50 = 2818.38 nM T20709 CDB83R 17516658 EC50 > 30000 nM T20709 CS2PX9 18204435 EC50 = 570 nM T20709 CLGM48 19571628 EC50 = 562 nM T20709 C7T8JC 19958494 Ki > 10000 nM T20709 C6LI5E 19958507 Ki > 10000 nM T20709 C3T5HF 21509921 Ki > 10000 nM T20709 CBN84K 22065997 Ki > 10000 nM T20709 C5WCD3 22745278 EC50 = 9.1 nM T20709 CXCO68 24192587 Ki = 676 nM T20709 CY21RE 24841480 Ki = 54 nM T20709 C4SY8G 24846938 Ki = 1.49 nM T20709 CF26NI 24865894 EC50 = 2818.38 nM T20709 C9YN3A 24894514 Ki = 56234.13 nM T20709 C8ND1U 24894515 Ki = 79432.82 nM T20709 CX2HR8 24894516 Ki = 47863.01 nM T20709 CG4B9R 24894624 Ki = 21379.62 nM T20709 C7KF9R 24894626 Ki = 5128.61 nM T20709 CFA60S 24894627 Ki = 6456.54 nM T20709 CT8B3K 24894629 Ki = 4365.16 nM T20709 CMF04K 24894631 Ki = 69183.1 nM T20709 CP08SJ 24894632 Ki = 24547.09 nM T20709 CLJK58 24894633 Ki = 58884.37 nM T20709 CR86FA 24894634 Ki = 28183.83 nM T20709 C9J3NX 24894636 Ki = 13803.84 nM T20709 CR7D1L 24967746 EC50 = 12.59 nM T20709 C8IXC0 24979170 EC50 = 3800 nM T20709 C5MYC3 25010776 EC50 > 30000 nM T20709 C18VYH 25015647 EC50 > 40000 nM T20709 CA20NZ 25025581 Ki = 251.19 nM T20709 CBY3O2 25070582 IC50 = 300 nM T20709 CXBF68 25110764 EC50 > 50000 nM T20709 C50IKG 25110765 EC50 > 50000 nM T20709 CK0BT7 25147647 Ki = 6606.93 nM T20709 CF0A4M 25162692 EC50 = 1584.89 nM T20709 CE2OG1 25199525 EC50 = 125.89 nM T20709 CRFJ43 25207745 EC50 = 794.33 nM T20709 CP2T6G 25230693 EC50 = 199.53 nM T20709 CAH1Y5 26441386 EC50 = 1698.24 nM T20709 CHY2N1 29262717 EC50 = 1100 nM T20709 CIHF79 30270932 EC50 = 389.05 nM T20709 C7IO6Q 30299339 EC50 = 850 nM T20709 C5M0FU 41358726 EC50 = 2100 nM T20709 C7P5XV 41528344 EC50 = 2700 nM T20709 C45ZNS 42596928 Ki = 2.63 nM T20709 C5DC7E 42598357 EC50 = 794.33 nM T20709 CO6QB0 42598358 EC50 = 100 nM T20709 CDPA93 42598359 EC50 = 1584.89 nM T20709 CAM5P6 42598360 EC50 = 158.49 nM T20709 C58SRK 42598586 EC50 = 1584.89 nM T20709 CYL45Z 42598591 EC50 = 39.81 nM T20709 C6S2HI 42598828 EC50 = 199.53 nM T20709 C2GYA4 42598829 EC50 = 501.19 nM T20709 C5CZ7P 42599068 EC50 = 158.49 nM T20709 C7O2ZV 42599070 EC50 = 31.62 nM T20709 C6BUZ5 42599071 EC50 = 501.19 nM T20709 C69BGH 43988968 EC50 > 10000 nM T20709 CD75UN 43989253 EC50 = 1122.02 nM T20709 CRQ2X4 43989254 EC50 > 10000 nM T20709 CS40ML 44123747 IC50 > 10000 nM T20709 C2AV1K 44190762 IC50 = 1340 nM T20709 CMR7T1 44204999 EC50 > 25118.86 nM T20709 C6GXL0 44208359 EC50 = 300 nM T20709 CGR6J0 44251556 EC50 > 30000 nM T20709 C2K0VZ 44253016 EC50 = 19.95 nM T20709 C2LFH7 44274302 Ki = 12302.69 nM T20709 CZX4M3 44274317 Ki = 33884.42 nM T20709 C5L3FV 44274400 Ki = 21379.62 nM T20709 CF47ZS 44274417 Ki = 46773.51 nM T20709 CCK63Z 44274432 Ki = 54954.09 nM T20709 CZ1U0E 44274433 Ki = 24547.09 nM T20709 C3XP7C 44274441 Ki = 12589.25 nM T20709 CO1RL0 44274468 Ki = 22387.21 nM T20709 C9JX7D 44274469 Ki = 12022.64 nM T20709 CF36IC 44274477 Ki = 89125.09 nM T20709 CC2OD4 44278111 Ki > 10000 nM T20709 CRMA84 44278114 Ki > 10000 nM T20709 CF0Y4M 44278115 Ki > 10000 nM T20709 C9Z0LT 44299564 Ki = 794.33 nM T20709 CX28HR 44299589 Ki = 1000 nM T20709 CPL36O 44299599 Ki = 1949.84 nM T20709 CFN95A 44299616 Ki = 891.25 nM T20709 CE4L1V 44299635 Ki = 1737.8 nM T20709 C6WG2J 44301710 Ki = 4.365 nM T20709 C9TWN3 44302727 IC50 = 6027.8 nM T20709 C5S8UL 44302728 IC50 = 301.1 nM T20709 CQ4B5T 44302741 IC50 = 359.6 nM T20709 C0AZF5 44302755 IC50 = 1498.3 nM T20709 CR5T1J 44302775 IC50 = 1624 nM T20709 CY8PD1 44302776 IC50 = 464.8 nM T20709 C7GY5J 44302788 IC50 = 501 nM T20709 CAV72D 44302793 IC50 = 4741.3 nM T20709 CV9QM6 44302813 IC50 = 3713.8 nM T20709 C43QTF 44302833 IC50 = 1474.8 nM T20709 CF74EQ 44302834 IC50 = 2633.7 nM T20709 C6J3EY 44302879 IC50 = 9927.5 nM T20709 CIU20B 44302900 IC50 = 2050 nM T20709 CGNA91 44302901 IC50 = 9735.2 nM T20709 C1RGS9 44304818 Ki = 7900 nM T20709 CVX13Q 44318736 Ki = 48 nM T20709 CT58BQ 44318766 Ki = 840 nM T20709 CR2T3J 44318817 Ki = 960 nM T20709 CL0HY5 44318929 Ki = 42 nM T20709 C01CVA 44318930 Ki = 300 nM T20709 C5VLY2 44326733 Ki = 24000 nM T20709 CSK4B0 44346542 IC50 = 2030 nM T20709 CU2X1V 44356367 IC50 = 8000 nM T20709 C7YTV9 44385809 Ki = 74 nM T20709 CHD9O7 44386115 Ki = 60 nM T20709 C1B4QL 44403095 Ki > 10000 nM T20709 C1YL7Z 44403098 Ki > 10000 nM T20709 CFV98A 44403101 Ki > 10000 nM T20709 C6OY9S 44403102 Ki > 10000 nM T20709 CH4SX6 44403105 Ki > 10000 nM T20709 C12FIH 44403106 Ki > 10000 nM T20709 C4LKC1 44404394 Ki > 10000 nM T20709 C3EJ4G 44404396 Ki > 10000 nM T20709 C6GLV1 44408714 Ki = 9120.11 nM T20709 C4QTI3 44415886 Ki = 180 nM T20709 CC9AV3 44418764 Ki = 25.12 nM T20709 CV6UQ3 44419370 Ki > 100000 nM T20709 C2N5LX 44422691 EC50 = 2511.89 nM T20709 CIRB78 44422696 Ki = 45708.82 nM T20709 CHT24X 44422698 EC50 = 25118.86 nM T20709 CDE8A1 44428745 Ki = 40.74 nM T20709 CG45PO 44437242 Ki = 682 nM T20709 C6I2JO 44437248 Ki = 5932 nM T20709 CZI05O 44437258 Ki = 5986 nM T20709 C7VP1Y 44437297 Ki = 1681 nM T20709 C5GT7C 44437302 Ki > 10000 nM T20709 C37QFT 44437307 Ki = 2265 nM T20709 CRC2Y5 44439387 Ki = 42000 nM T20709 C3ZT7I 44439388 Ki = 78000 nM T20709 CKU9N8 44439389 Ki = 70000 nM T20709 C20VDP 44439390 Ki = 18000 nM T20709 C6RKA9 44439391 Ki = 12000 nM T20709 CI9D7G 44439392 Ki = 94000 nM T20709 CDE27X 44439393 Ki = 95000 nM T20709 CIQW67 44439394 Ki = 68000 nM T20709 CV93LJ 44439395 Ki > 300000 nM T20709 CPX5Q2 44439396 Ki = 1400 nM T20709 C2R0SX 44439397 Ki = 50000 nM T20709 C4CMV7 44439398 Ki = 200 nM T20709 C8YQ4P 44439399 Ki = 200 nM T20709 C6YA9O 44439400 Ki = 12000 nM T20709 C89ZPX 44439401 Ki = 2000 nM T20709 CE60JL 44439402 Ki = 2800 nM T20709 C65GSE 44439403 Ki = 200 nM T20709 CKUG90 44439404 Ki = 1600 nM T20709 CTYP87 44439405 Ki = 700 nM T20709 C3UBA6 44439406 Ki = 11000 nM T20709 C7HV8X 44439407 Ki = 4500 nM T20709 CD4T3S 44439408 Ki = 300 nM T20709 C07XPE 44439409 Ki = 4500 nM T20709 CMU43Q 44439410 Ki = 19000 nM T20709 C36LXN 44446840 Ki = 87096.36 nM T20709 C6S4XU 44448379 Ki = 2691.53 nM T20709 C0ZLX8 44448383 Ki = 12.59 nM T20709 C1USW7 44448418 Ki = 11220.18 nM T20709 C8NB9P 44448421 Ki = 74.13 nM T20709 CMF5E6 44448456 Ki = 11220.18 nM T20709 CH9IC4 44448495 Ki = 22908.68 nM T20709 CHAX49 44448499 Ki = 1230.27 nM T20709 CA9QL5 44448537 Ki = 4786.3 nM T20709 CJK41H 44448645 Ki = 288.4 nM T20709 C12XGE 44456400 Ki > 10000 nM T20709 CVA67X 44568347 Ki = 21 nM T20709 CY9C2A 44571572 Ki > 100000 nM T20709 CM0D1J 44575653 IC50 = 10 nM T20709 CN68YI 44578707 Ki = 2454.71 nM T20709 CHUN40 44578928 EC50 > 50000 nM T20709 CZYP06 44578975 EC50 > 50000 nM T20709 CCIT12 44578976 EC50 > 50000 nM T20709 CW53ZF 44578977 EC50 > 50000 nM T20709 CYHM34 44578978 EC50 > 50000 nM T20709 CGF7A4 44579375 EC50 > 50000 nM T20709 C1OCB6 44579416 EC50 > 50000 nM T20709 CARW17 44579417 EC50 > 50000 nM T20709 C2DFV7 44579418 EC50 > 50000 nM T20709 CTC8H6 44579419 EC50 > 50000 nM T20709 CYR0O3 44579457 EC50 > 50000 nM T20709 CF1EA4 44579458 EC50 > 50000 nM T20709 CQ4Y8O 44589531 EC50 > 30000 nM T20709 CL40CM 44589593 EC50 > 30000 nM T20709 CKS5V4 44589594 EC50 > 30000 nM T20709 CXB30W 44589595 EC50 > 30000 nM T20709 CM5LJ8 44589596 EC50 > 30000 nM T20709 CPXE19 44589643 EC50 > 30000 nM T20709 C8AJO6 44589644 EC50 > 30000 nM T20709 CFS1A4 44589645 EC50 > 30000 nM T20709 C71EHI 44589646 EC50 > 30000 nM T20709 CQB5A9 44589681 EC50 = 9.1 nM T20709 CUA62X 44593616 Ki = 316.23 nM T20709 CN9ID8 44593617 Ki = 407.38 nM T20709 CDM56I 44593618 Ki = 42.66 nM T20709 CU63PQ 44593619 Ki = 33.11 nM T20709 CL8D2S 44593620 Ki = 93.33 nM T20709 CI97KQ 44593621 Ki = 501.19 nM T20709 CL5O8E 44602489 EC50 > 30000 nM T20709 CH2Z3O 44610056 Ki = 0.35 nM T20709 CVZ6Y1 44627739 Ki = 104.71 nM T20709 CE6A9F 44627740 Ki = 14.13 nM T20709 C6EU7P 44627741 Ki = 158.49 nM T20709 CW40TR 44627742 Ki = 77.62 nM T20709 C5GIU6 44627743 Ki = 64.57 nM T20709 CK9DO1 44627745 Ki = 15.49 nM T20709 CJ8S1L 44627747 Ki = 38.02 nM T20709 C5LY8C 44627851 Ki = 19.5 nM T20709 CC4A3X 44627853 Ki = 3.981 nM T20709 CH4N5J 44627854 Ki = 54.95 nM T20709 CO8C6D 44627855 Ki = 549.54 nM T20709 COL8E1 44627856 Ki = 3090.3 nM T20709 C6WS7M 44627857 Ki = 4.266 nM T20709 C43BJY 44627859 Ki = 33.11 nM T20709 CW0X6A 44627955 Ki = 371.54 nM T20709 CXNF31 44627957 Ki = 2344.23 nM T20709 C4LOY2 45115589 Ki < 1000 nM T20709 CY1O9Z 45142486 EC50 = 95 nM T20709 C9U0VH 45259185 Ki = 281.84 nM T20709 CNC1R2 45259186 Ki = 104.71 nM T20709 CP2CZ7 45259187 Ki = 316.23 nM T20709 CW14TS 45259188 Ki = 15.85 nM T20709 CO8W1X 45259189 Ki = 19.05 nM T20709 CF16YZ 45259190 Ki = 112.2 nM T20709 C7L1CU 45266348 Ki = 95.5 nM T20709 C2N9UV 45501061 EC50 = 897 nM T20709 CC18GX 45501063 EC50 = 588.84 nM T20709 CRE46S 45501064 EC50 = 616.6 nM T20709 CU4V5R 46227410 Ki > 100000 nM T20709 CWQ1L9 46227412 Ki = 30902.95 nM T20709 CX2E6A 46227414 Ki > 100000 nM T20709 C0Z4RD 46227416 Ki > 100000 nM T20709 CK2R5G 46227454 Ki > 100000 nM T20709 C8OZI6 46227456 Ki = 44668.36 nM T20709 CB45NM 46227458 Ki > 100000 nM T20709 C1J0IF 46227460 Ki = 57543.99 nM T20709 CQ4DI6 46227480 Ki = 87096.36 nM T20709 CHKL80 46227482 Ki = 25703.96 nM T20709 CVP7T6 46227484 Ki = 30199.52 nM T20709 CC6RH5 46227486 Ki = 53703.18 nM T20709 CSQ0V3 46227554 Ki = 93325.43 nM T20709 C1Q0MH 46830362 IC50 = 1500 nM T20709 CH3ID7 46830363 IC50 = 3700 nM T20709 C01YTE 46871665 IC50 = 1584.89 nM T20709 CUY51M 46871666 IC50 = 3162.28 nM T20709 CYLZ50 46871844 IC50 = 158.49 nM T20709 CCZ5I8 46883796 IC50 = 3700 nM T20709 CVCF68 46883843 IC50 > 10000 nM T20709 CW70YU 46890977 IC50 = 398.11 nM T20709 CJ74AZ 46891076 IC50 = 7943.28 nM T20709 CTSZ49 46891179 IC50 = 3162.28 nM T20709 COT8S4 46891375 EC50 > 10000 nM T20709 CW1YX7 46891488 IC50 = 5011.87 nM T20709 CB1Z5A 46905390 IC50 = 534.5 nM T20709 C67XQI 46945663 EC50 > 30000 nM T20709 CT8MX0 49663929 IC50 = 650 nM T20709 C7IAW9 49663949 IC50 = 346.74 nM T20709 CD39WZ 49665121 IC50 > 10000 nM T20709 C7QVN3 49671356 IC50 = 530 nM T20709 CIR1Z3 49674582 EC50 = 645.65 nM T20709 C2LZJ0 49783209 Ki = 760 nM T20709 C57SMG 49783415 Ki = 2579 nM T20709 C0TG6I 49783419 Ki > 10000 nM T20709 C20SCO 49797320 Ki = 5478 nM T20709 C29QSB 49797322 Ki = 792 nM T20709 CT4QU7 49797325 Ki = 6041 nM T20709 C7ROA4 49797387 Ki = 1174.9 nM T20709 CQX3I5 49797388 Ki = 616.6 nM T20709 C9VG5A 49797390 Ki = 162181.01 nM T20709 C6RES8 49797391 Ki = 22387.21 nM T20709 C2E0DY 49797392 Ki = 100000 nM T20709 CLF8X5 49797394 Ki = 9772.37 nM T20709 CXD65I 49797395 Ki = 1174.9 nM T20709 CPI6N0 49853777 IC50 > 100000 nM T20709 C94GDK 49853778 IC50 > 100000 nM T20709 CHV3U8 49853881 IC50 > 100000 nM T20709 CTBY97 49853883 IC50 > 100000 nM T20709 CQP63D 49853884 IC50 = 73000 nM T20709 CY8M9A 49853885 IC50 > 100000 nM T20709 CN0JU9 49853987 IC50 > 100000 nM T20709 C8DVX6 49855131 IC50 > 100000 nM T20709 C2RY0J 50878551 Ki > 10000 nM T20709 C1W6TV 50898777 Ki > 10000 nM T20709 CXMZ73 50898778 Ki > 10000 nM T20709 CE4KP1 51050257 Ki > 10000 nM T20709 C1ZT0O 52176746 IC50 = 6080 nM T20709 CM47HJ 52176747 IC50 = 426.58 nM T20709 C2CI4N 53002537 EC50 = 6309.57 nM T20709 C5F0HW 53002540 EC50 = 1412.54 nM T20709 CZW9T0 53002564 EC50 = 562.34 nM T20709 C6KU3Z 53303986 IC50 = 3100 nM T20709 CR4W9L 53324553 Ki = 705 nM T20709 CO3RX1 53382478 EC50 = 1737.8 nM T20709 CAG82Y 53382480 EC50 = 154.88 nM T20709 CPHK81 53382482 EC50 = 80 nM T20709 C6WK9C 53382484 EC50 = 269.15 nM T20709 CJ13RP 53382492 EC50 = 249 nM T20709 CPW56J 53382493 EC50 = 1410 nM T20709 CM3N6F 53382497 EC50 = 294 nM T20709 C2DG9B 53382498 EC50 = 52 nM T20709 C53WVJ 53382500 EC50 = 1370 nM T20709 CP7E2L 53382502 EC50 = 323.59 nM T20709 CGJD69 53382503 EC50 = 810 nM T20709 CAP95B 53382504 EC50 = 104 nM T20709 CE1X7K 53382505 EC50 = 128 nM T20709 CYN8A7 53382508 EC50 = 208 nM T20709 CTNM37 53382512 EC50 = 107 nM T20709 C86DNC 53382513 EC50 = 416.87 nM T20709 CQX56E 53382515 EC50 = 307 nM T20709 COA3J9 53382516 EC50 = 669 nM T20709 CDRZ30 53382518 EC50 = 123.03 nM T20709 CT2Z4Y 53382520 EC50 = 600 nM T20709 CVH48U 53382522 EC50 > 30000 nM T20709 CS1OI7 53382523 EC50 = 56 nM T20709 C9ZX8K 53382524 EC50 = 61 nM T20709 C8KUR9 53382526 EC50 = 288.4 nM T20709 CCIH19 53382528 EC50 = 107.15 nM T20709 CMG92P 53382529 EC50 = 147 nM T20709 C7CZ2M 53382530 EC50 = 30000 nM T20709 CMRT42 53382534 EC50 = 1995.26 nM T20709 C8ILE5 53382540 EC50 = 354.81 nM T20709 CZBV95 53382541 EC50 = 926 nM T20709 CWR16G 53382542 EC50 = 77 nM T20709 C3DW2N 53382544 EC50 = 844 nM T20709 C7YP3A 53385782 EC50 > 10000 nM T20709 CMOZ61 53475319 Ki = 2279 nM T20709 C30MNL 55485382 EC50 = 6165.95 nM T20709 CNG41A 55661332 EC50 = 954.99 nM T20709 CJ3C9G 56592900 EC50 > 10000 nM T20709 C2PFE9 56592902 EC50 > 10000 nM T20709 CH4A1V 56592905 EC50 = 2344.23 nM T20709 C9RW1B 56592910 EC50 = 1288.25 nM T20709 CAT12I 56592911 EC50 = 7762.47 nM T20709 CR46HD 56592923 EC50 > 10000 nM T20709 CWI81F 56592928 EC50 > 10000 nM T20709 C4NGA8 56592929 EC50 > 10000 nM T20709 CT14BV 56592932 EC50 = 7079.46 nM T20709 CQ0H9L 56592943 EC50 > 10000 nM T20709 C8WHT5 56593934 Ki = 10000 nM T20709 CU0NE5 56672197 Ki = 1364 nM T20709 CB0P9N 56944383 Ki > 1000 nM T20709 C1TC7Q 56963799 Ki = 415 nM T20709 C3WC7Z 56965018 Ki = 4.898 nM T20709 CUP4Y0 57326139 Ki = 25118.86 nM T20709 C1G9XY 57326141 Ki > 100000 nM T20709 CG3YS9 57326143 Ki = 12302.69 nM T20709 CCYU25 57326145 Ki = 29512.09 nM T20709 CS86GL 57326232 Ki = 151.36 nM T20709 C3AF0Z 57326234 Ki = 1.479 nM T20709 CLSW35 57326236 Ki = 11220.18 nM T20709 CL3R5D 57326238 Ki = 16982.44 nM T20709 C4G1LB 57326325 Ki = 70.79 nM T20709 C6CB9J 57326326 Ki = 2.344 nM T20709 C5OJP0 57391102 EC50 > 30000 nM T20709 C17GMJ 57393065 IC50 > 30000 nM T20709 C6HBG0 57396813 IC50 = 4800 nM T20709 CQ5BG6 57525860 EC50 > 30000 nM T20709 C9TMZ3 57558000 Ki > 100000 nM T20709 C6IJ2F 57664418 Ki = 194.98 nM T20709 CA14SG 58653718 Ki > 100000 nM T20709 CRV9X7 59654579 EC50 = 115 nM T20709 CAZ9B3 62705488 IC50 > 10000 nM T20709 C9F4JW 62705832 IC50 > 10000 nM T20709 CA5FP7 66561966 Ki = 6167 nM T20709 C3XL7O 66561967 Ki = 1098 nM T20709 CCB1T5 68764898 Ki = 865 nM T20709 CF8DC9 70681307 Ki = 15.85 nM T20709 CXT67P 70683405 Ki = 18.62 nM T20709 CN98LU 70685504 Ki = 12.3 nM T20709 CT41UM 70687661 Ki = 12.88 nM T20709 CJLS94 71449148 Ki = 12.74 nM T20709 C9VZ8J 71450550 Ki = 685 nM T20709 CY3M8B 71451570 IC50 = 140 nM T20709 C4NDR3 71452382 Ki = 470 nM T20709 CYK20Z 71452384 Ki = 2961 nM T20709 CDTW09 71452387 Ki = 1302 nM T20709 C5WK8L 71452756 Ki = 0.09 nM T20709 CK81FI 71452793 Ki = 15.2 nM T20709 CX26PA 71454562 Ki = 45.05 nM T20709 CX35MW 71454563 Ki = 0.32 nM T20709 C6G2HC 71455894 Ki = 1233 nM T20709 CFBC49 71455896 Ki = 8135 nM T20709 CVI7S2 71457690 Ki = 1118 nM T20709 CP7JI0 71457691 Ki = 514 nM T20709 C5DLQ2 71459553 Ki > 10000 nM T20709 CK5T4P 71459604 Ki = 977 nM T20709 COQ67L 71459971 Ki = 18.4 nM T20709 C2OIW1 71461631 IC50 = 145.4 nM T20709 CG8F1C 71461681 Ki = 17.9 nM T20709 CL91AC 71463022 Ki = 2871 nM T20709 CKX5O8 71463061 Ki = 2338 nM T20709 C1Y9IC 71463063 Ki = 659 nM T20709 CKT3C6 71516707 EC50 > 10000 nM T20709 CV24CP 71518072 EC50 > 30000 nM T20709 CG7HA3 71528087 EC50 = 15 nM T20709 CCVD76 71528088 EC50 = 320 nM T20709 CE82HN 71533671 EC50 = 13 nM T20709 C68UAI 71574174 Ki > 100000 nM T20709 C3MJ7B 71575027 Ki = 11500 nM T20709 CN82HY 71575122 Ki = 10500 nM T20709 CY1Q9O 71575447 Ki = 1890 nM T20709 CNS4V8 71575552 Ki > 100000 nM T20709 CM9SQ2 71575553 Ki > 100000 nM T20709 C89MPL 71575652 Ki = 5740 nM T20709 CM8UN7 71598549 IC50 > 30000 nM T20709 C1OE9J 71607097 IC50 > 30000 nM T20709 CEIH75 71683155 EC50 = 58.88 nM T20709 C6YQ4H 71719475 EC50 = 29 nM T20709 C3FQY2 71806339 IC50 > 10000 nM T20709 CHE5O6 72545089 Ki > 100000 nM T20709 CI6D4E 72545091 Ki > 100000 nM T20709 CKFW54 72545094 Ki > 100000 nM T20709 CWLO54 72545096 Ki > 100000 nM T20709 C5D4PA 72545098 Ki > 100000 nM T20709 CR39AG 72545326 Ki > 100000 nM T20709 C5HLF7 72545329 Ki > 100000 nM T20709 CL9C0F 72713879 EC50 = 560 nM T20709 CPQW85 72713884 EC50 = 309.03 nM T20709 CP3M0S 72714095 EC50 = 575.44 nM T20709 CUR3P7 72714096 EC50 = 140 nM T20709 CN32ZF 72714097 EC50 = 100 nM T20709 CCGM95 72714098 EC50 = 346.74 nM T20709 C5ZJ1Y 72714099 EC50 = 239.88 nM T20709 C6ZA8H 72945087 EC50 = 47 nM T20709 CC65OA 73213195 Ki > 10000 nM T20709 CW83DK 73213196 Ki > 10000 nM T20709 C46HUP 73345823 Ki = 89.6 nM T20709 CRG9J8 73346332 Ki = 4038 nM T20709 CK0HR9 73346334 Ki = 892 nM T20709 C6J0TM 73346336 Ki = 619 nM T20709 C5G3YO 73346357 EC50 = 104.71 nM T20709 CY60RD 73347826 Ki = 1302 nM T20709 CC35AI 73347827 Ki = 2796 nM T20709 C27EIP 73347857 EC50 = 128.82 nM T20709 CY2IB5 73349362 Ki = 3904 nM T20709 CI4U3P 73349391 EC50 = 125.89 nM T20709 C58SJG 73349591 Ki > 100000 nM T20709 CA6Z1P 73349592 Ki > 100000 nM T20709 C8GQK9 73350823 Ki = 1270 nM T20709 CDS4F1 73350931 Ki = 1265 nM T20709 CH2B4Y 73350932 Ki = 7385 nM T20709 C4RCZ0 73350962 EC50 = 130 nM T20709 CA8L9Y 73351145 Ki > 100000 nM T20709 CV1U7L 73352414 Ki = 707 nM T20709 C87LGB 73352415 Ki = 3586 nM T20709 CFM9Z0 73353378 Ki = 285 nM T20709 C1NJ0R 73353884 Ki = 6528 nM T20709 CZ65RX 73353907 EC50 = 218.78 nM T20709 C4F7VK 73355415 Ki = 354 nM T20709 CA4CP6 73355416 Ki = 6993 nM T20709 C81CIL 73355418 Ki = 6806 nM T20709 C3Z5LT 73355419 Ki = 3809 nM T20709 C10ASZ 73355420 Ki = 5908 nM T20709 C2K5DS 73672762 EC50 = 93 nM T20709 CHV3W1 73774630 EC50 = 91 nM T20709 C7G0UH 75203027 EC50 = 260 nM T20709 C8IDL3 75306277 Ki > 1000 nM T20709 C43NME 76313419 IC50 > 10000 nM T20709 C5JNZ1 76324306 IC50 > 10000 nM T20709 CXKN87 78319052 EC50 = 11 nM T20709 CP1AM5 86292822 EC50 = 60 nM T20709 CNW34R 87057213 EC50 = 690 nM T20709 C04VWL 87057214 EC50 = 620 nM T20709 CX8Y6K 87057216 EC50 = 40 nM T20709 C8W5QT 89445225 EC50 = 1100 nM T20709 C0HGV9 89445242 EC50 = 1000 nM T20709 COLZ67 89445250 EC50 = 2200 nM T20709 C7JW0B 89445258 EC50 = 2000 nM T20709 CL7NM6 89452242 EC50 = 120 nM T20709 CR0EY3 89452445 EC50 = 230 nM T20709 CHT03L 89452615 EC50 > 10000 nM T20709 C7OU9P 89452686 EC50 = 1200 nM T20709 CZ3M2U 89452852 EC50 > 10000 nM T20709 C2BM9L 89768534 EC50 = 251 nM T20709 CB4Y7R 89768546 EC50 = 549.54 nM T20709 C4ST8E 89768704 EC50 = 436.52 nM T20709 CMFP38 89768734 EC50 = 1047 nM T20709 CTOR31 89768736 EC50 = 208.93 nM T20709 CJ27OR 89768749 EC50 = 181.97 nM T20709 CZ3N8B 89777032 EC50 = 416.87 nM T20709 CYX9R8 89777050 EC50 = 72 nM T20709 CN0R6C 89777060 EC50 = 22.39 nM T20709 CB52US 89777104 EC50 = 63.1 nM T20709 CT3ZV4 89777143 EC50 = 60.2 nM T20709 C2N5PF 89777146 EC50 = 602.56 nM T20709 C5T3DH 89777147 EC50 = 177.83 nM T20709 C5MR9K 89777151 EC50 = 91 nM T20709 C4NVC7 89777179 EC50 = 33.11 nM T20709 CA4EH5 89777192 EC50 = 363 nM T20709 CUFI32 89777224 EC50 = 2238.72 nM T20709 CX29WN 89777226 EC50 = 23.99 nM T20709 CKO0Z3 89777237 EC50 = 217 nM T20709 CQ0IM3 89777238 EC50 = 354.81 nM T20709 C7WOC3 89777239 EC50 = 80 nM T20709 C54MXA 89777257 EC50 = 295.12 nM T20709 CRZ34V 89777258 EC50 = 26.92 nM T20709 C80GHA 89777261 EC50 = 363 nM T20709 CCEI47 89777262 EC50 = 1584.89 nM T20709 C6JE1I 89777266 EC50 = 150 nM T20709 C5TQD1 89777269 EC50 = 263.03 nM T20709 CP42GR 89777270 EC50 = 446.68 nM T20709 CJ3DU4 89777274 EC50 = 562.34 nM T20709 C8HV2O 89777316 EC50 = 144 nM T20709 CPJ24Q 89777355 EC50 = 177.83 nM T20709 C3MFV0 89777356 EC50 = 24.55 nM T20709 CZ58KT 89777437 EC50 = 63.1 nM T20709 C8LPG4 89777449 EC50 = 316 nM T20709 C5S4PX 89777463 EC50 = 48.98 nM T20709 C5WQ7P 89777468 EC50 = 83.18 nM T20709 C6FIV0 89777513 EC50 = 776.25 nM T20709 C4RUP2 101882890 Ki = 1.072 nM T20709 C9O0PU 117910878 EC50 = 1500 nM T20709 CZ53PE 117916853 EC50 = 5100 nM T20709 CSZ87Q 117916866 EC50 = 5900 nM T20709 CY92QJ 117916869 EC50 > 10000 nM T20709 CFP2H7 117916889 EC50 = 1500 nM T20709 CWE1K6 117916898 EC50 = 6400 nM T20709 CSDI45 117916916 EC50 = 2700 nM T20709 CAR0M7 117917122 EC50 > 10000 nM T20709 CQI38V 117917123 EC50 = 5600 nM T20709 C2OJ6W 117917124 EC50 = 2100 nM T20709 CC3YS5 118706050 Ki > 100000 nM T20709 C6DXV9 118706052 Ki > 100000 nM T20709 CL4EO9 118706054 Ki = 20892.96 nM T20709 C4JY5S 118719502 IC50 > 30000 nM T20709 CI8CR0 118719920 Ki = 26.3 nM T20709 CV1WX5 118719921 Ki = 7.943 nM T20709 CIAG59 118719922 Ki = 0.8913 nM T20709 CC5Q8Y 118719923 Ki = 6.607 nM T20709 CC8R6U 118719924 Ki = 14.45 nM T20709 CT8KO4 118719925 Ki = 588.84 nM T20709 C16DHZ 118719926 Ki = 446.68 nM T20709 CLA06I 118719927 Ki = 389.05 nM T20709 CF20SR 118719928 Ki = 154.88 nM T20709 C6N7HV 118719929 Ki = 112.2 nM T20709 C64BIA 118719930 Ki = 95.5 nM T20709 CG4ZV5 118719931 Ki = 32.36 nM T20709 C05OBV 118723724 Ki > 100000 nM T20709 C5LF3X 121053081 IC50 = 5370.32 nM T20709 CO23UE 121053110 IC50 = 1258.93 nM T20709 CKEJ96 121053122 IC50 = 407.38 nM T20709 CKP85M 122189495 EC50 = 235 nM T20709 C2H3QF 122189496 EC50 = 393 nM T20709 C9HG5K 122189499 EC50 = 113 nM T20709 CAJ45R 122190994 EC50 = 1110 nM T20709 C7TL4G 122191001 EC50 = 355 nM T20709 CA02ZK 122191002 EC50 = 227 nM T20709 C80JRU 122191004 EC50 = 1360 nM T20709 CF8N0T 122191005 EC50 = 3720 nM T20709 CR93HM 122191007 EC50 = 392 nM T20709 CRF36I 122191008 EC50 = 405 nM T20709 CQX7P1 122195090 EC50 = 86 nM T20709 CSG15Z 122387444 Ki = 2691.53 nM T20709 C8LEC0 122387446 Ki = 520 nM T20709 CB3WR0 122387447 Ki = 1659.59 nM T20709 CYG57C 122387448 Ki = 4265.8 nM T20709 CKCV39 122387449 Ki = 3162.28 nM T20709 C3D2XL 127043450 EC50 = 1862.09 nM T20709 C7WI3E 127043631 EC50 = 812.83 nM T20709 C7NQX2 127043632 EC50 = 4365.16 nM T20709 CC6DY3 127043635 EC50 = 600 nM T20709 C3E1RN 127043636 EC50 = 1737.8 nM T20709 CGS8B3 127043637 EC50 = 2290.87 nM T20709 CVL05H 127043638 EC50 = 690 nM T20709 CK8VE4 127043639 EC50 = 1047.13 nM T20709 CJ2O5A 127044078 EC50 = 575.44 nM T20709 CQN0X5 127044525 EC50 = 4265.8 nM T20709 C0JV8P 127044539 EC50 = 970 nM T20709 C4DIY3 127044706 EC50 = 1174.9 nM T20709 CSX3N2 127045035 IC50 = 1500 nM T20709 CART92 127045185 IC50 = 2400 nM T20709 CW4O0Z 129277684 EC50 = 14 nM T20709 C9MI5R 129277689 EC50 = 17 nM T20709 CJ94GK 129316454 EC50 > 10000 nM T20709 CT81OY 132060776 Ki = 2681 nM T20709 C56GQW 132063677 EC50 = 281.84 nM T20709 CAVB41 132584404 Ki > 10000 nM T20709 CBU81N 134149168 Ki > 10000 nM T20709 CNTC06 134207678 EC50 = 12 nM T20709 C91CGP 134207679 EC50 = 84 nM T20709 CN5XM4 134207680 EC50 = 60 nM T20709 CTW7F4 134207681 EC50 = 1900 nM T20709 C08GLT 134207682 EC50 = 140 nM T20709 CU2JC6 134207684 EC50 = 300 nM T20709 CIRG09 134207685 EC50 = 2000 nM T20709 CJF0E1 134207687 EC50 = 89 nM T20709 COT7F6 134207689 EC50 = 620 nM T20709 CY24XH 134207690 EC50 = 120 nM T20709 CQNK23 134207694 EC50 = 160 nM T20709 C2X6BZ 134207697 EC50 = 110 nM T20709 C6DVO4 134207699 EC50 = 130 nM T20709 C7S4DT 134207701 EC50 = 110 nM T20709 CP1R0B 134207702 EC50 = 160 nM T20709 C4QIG1 134207705 EC50 = 120 nM T20709 CTS04H 134207706 EC50 = 2100 nM T20709 CSVR09 134207707 EC50 = 12 nM T20709 CT4L6M 134207710 EC50 = 240 nM T20709 CQA8K6 134207711 EC50 = 26 nM T20709 CMPD81 134207712 EC50 = 270 nM T20709 CQW1R2 134207713 EC50 = 16 nM T20709 CPO71C 134207717 EC50 = 120 nM T20709 C2LW6M 134207719 EC50 = 46 nM T20709 CS59OL 134207720 EC50 = 8 nM T20709 CI0DP2 134207721 EC50 = 20 nM T20709 C43DAS 134207723 EC50 = 17 nM T20709 CMQ04E 134207724 EC50 = 250 nM T20709 CL18ED 134207726 EC50 = 22 nM T20709 CLGD37 134207727 EC50 = 310 nM T20709 CA16JM 134207728 EC50 = 140 nM T20709 CQ62MV 134207729 EC50 = 410 nM T20709 CU3CF4 134207730 EC50 = 1200 nM T20709 CB3WI5 134207731 EC50 = 270 nM T20709 C1CUF0 135150406 EC50 = 20 nM T20709 C1DNG0 135150478 EC50 = 20 nM T20709 C8Q3XO 135153778 EC50 = 22 nM T20709 CI82CJ 135153922 EC50 = 25 nM T20709 CH0RM5 135154300 EC50 = 18 nM T20709 CP75JB 135154593 EC50 = 20 nM T20709 C2MG0Y 135154616 EC50 = 14 nM T20709 CYV03R 135171475 EC50 = 18 nM T20709 C4OIU5 135171550 EC50 = 18 nM T20709 C4UX2M 135430667 Ki = 61.66 nM T20709 CIH0F3 137631537 EC50 = 8 nM T20709 C40FTE 137632597 EC50 = 208.93 nM T20709 C0AKV2 137632645 IC50 < 10000 nM T20709 CF91CJ 137632847 EC50 = 1548.82 nM T20709 C63CFB 137633344 EC50 = 616.6 nM T20709 CZ3F0B 137633670 IC50 < 10000 nM T20709 CO78XJ 137633999 EC50 = 54.95 nM T20709 CM5TH3 137634025 EC50 = 3162.28 nM T20709 CX0DA1 137634235 IC50 = 1000 nM T20709 CT4IG0 137634274 IC50 = 3981.07 nM T20709 CP07AG 137635043 EC50 = 18.62 nM T20709 CFHT72 137635323 IC50 = 501.19 nM T20709 CM9C1Z 137635723 EC50 = 91.2 nM T20709 C6QB9W 137635734 Ki = 5128.61 nM T20709 CVKN97 137635985 IC50 = 2398.83 nM T20709 CG7MC8 137636004 IC50 = 660.69 nM T20709 CX8O0V 137636308 Ki = 3162.28 nM T20709 CKX1C7 137636570 IC50 = 470 nM T20709 C26ECU 137636810 IC50 = 302 nM T20709 C54RXL 137637726 EC50 = 5370.32 nM T20709 C7VUW4 137637944 Ki = 10.3 nM T20709 CPVE08 137637971 IC50 = 520 nM T20709 CY8Q1V 137638270 Ki = 7.78 nM T20709 CL5FQ7 137638666 IC50 > 10000 nM T20709 C0YJ1N 137639216 IC50 = 2290.87 nM T20709 CWK2M3 137639344 IC50 = 691.83 nM T20709 CC2PK1 137640000 EC50 = 38.9 nM T20709 CZ4TA9 137640201 EC50 = 147.91 nM T20709 CX4A3N 137640511 Ki = 9332.54 nM T20709 C4AOR2 137640564 EC50 = 169.82 nM T20709 CKB8I3 137640923 IC50 = 562.34 nM T20709 CH6EU7 137640924 EC50 = 2951.21 nM T20709 C1F8UM 137641287 IC50 = 1122.02 nM T20709 CTR28H 137641641 EC50 = 213.8 nM T20709 CUDE96 137641843 IC50 = 1600 nM T20709 C19LSM 137641912 IC50 = 3310 nM T20709 C80CXI 137641943 EC50 = 102.33 nM T20709 C8I2AC 137642025 EC50 = 2041.74 nM T20709 CL2KH9 137642171 IC50 = 707.95 nM T20709 CN23BR 137642305 EC50 > 10000 nM T20709 C4Q6ZM 137642607 Ki = 1288.25 nM T20709 C9OEF1 137642731 IC50 = 77.62 nM T20709 C7G8UX 137643460 EC50 = 10.72 nM T20709 C9RBJ3 137643470 IC50 < 10000 nM T20709 CV3E1N 137644574 IC50 = 2884.03 nM T20709 C0KL6Q 137644962 Ki = 2630.27 nM T20709 C83CGS 137645044 EC50 = 933.25 nM T20709 CPCY48 137645406 Ki = 590 nM T20709 C1IVG4 137645408 EC50 = 1047.13 nM T20709 CO0X1G 137645473 EC50 = 27.54 nM T20709 CG8P6I 137645938 Ki = 575.44 nM T20709 CC2PL7 137646286 EC50 = 16.98 nM T20709 CJNU86 137646437 EC50 = 213.8 nM T20709 C85WCD 137646585 EC50 = 905 nM T20709 CTJ0G9 137646601 EC50 = 1659.59 nM T20709 CN4U1A 137646732 EC50 = 75.86 nM T20709 CJ6LK4 137647278 EC50 = 630.96 nM T20709 C4DQ7L 137647376 IC50 = 2380 nM T20709 CH3Q2R 137647522 IC50 = 407.38 nM T20709 C6W5ZT 137647620 EC50 = 165.96 nM T20709 C42SPH 137647679 IC50 = 940 nM T20709 C2XMK6 137647734 IC50 = 131.83 nM T20709 C5CU6F 137648177 IC50 = 302 nM T20709 CSAR57 137648504 IC50 = 2691.53 nM T20709 CKL75F 137649175 EC50 = 32.36 nM T20709 CKM30I 137649420 EC50 = 158.49 nM T20709 CW7QP6 137649829 IC50 = 194.98 nM T20709 CU73XZ 137650228 EC50 = 131.83 nM T20709 C0D5GL 137650247 EC50 = 33.11 nM T20709 CF04JU 137650402 EC50 = 229.09 nM T20709 CBN1K6 137650836 Ki = 3.631 nM T20709 C3CZX8 137651392 EC50 < 10000 nM T20709 C87IQK 137652430 EC50 = 489.78 nM T20709 CJYS30 137652916 EC50 > 10000 nM T20709 C3QNK9 137653138 EC50 = 147 nM T20709 C45VBZ 137653326 EC50 = 562.34 nM T20709 CL8S9G 137653452 EC50 = 50.12 nM T20709 C0WZ4D 137653550 IC50 = 90 nM T20709 CI71LV 137653737 EC50 = 870.96 nM T20709 C61WAG 137654353 IC50 = 323.59 nM T20709 C0YD5K 137654582 EC50 = 1288.25 nM T20709 C63FLU 137654912 EC50 < 10000 nM T20709 COA6N8 137654928 IC50 = 263.03 nM T20709 CWOV78 137655063 IC50 = 123.03 nM T20709 C5A2IW 137655194 IC50 > 10000 nM T20709 C2RMN5 137655354 IC50 = 1350 nM T20709 CP1LB3 137655482 IC50 > 10000 nM T20709 CUC54G 137655636 Ki = 199.53 nM T20709 CDB06R 137655902 IC50 = 229.09 nM T20709 C86GOA 137655967 IC50 = 2800 nM T20709 C3DLO5 137656219 EC50 = 28.84 nM T20709 CA5PM3 137656230 EC50 = 100 nM T20709 CNLM06 137656522 IC50 > 10000 nM T20709 CA9G1Z 137656749 EC50 = 2137.96 nM T20709 C46VBM 137656783 EC50 = 15.49 nM T20709 C7CDB6 137657309 EC50 = 933.25 nM T20709 C42IMG 137657888 EC50 = 562.34 nM T20709 CUNI94 137658023 IC50 = 169.82 nM T20709 C29ZBS 137658151 IC50 = 2570.4 nM T20709 CF4KQ3 137658248 IC50 = 117.49 nM T20709 C6TR7E 137658427 EC50 = 234.42 nM T20709 CL5MP1 137658662 EC50 = 18.2 nM T20709 C1L2MJ 137658887 IC50 < 10000 nM T20709 C1CG3Y 137659030 IC50 = 2570 nM T20709 CO2QM6 137659033 EC50 > 10000 nM T20709 CQN25D 137659727 EC50 = 74.13 nM T20709 CXV46L 137659754 IC50 = 510 nM T20709 CN19PG 137659901 EC50 = 1258.93 nM T20709 CK04TM 137660952 IC50 = 1330 nM T20709 C68QKL 137661317 Ki = 0.4677 nM T20709 CDA8V2 137661377 Ki = 1659.59 nM T20709 CZJS43 137661476 IC50 = 290 nM T20709 C1ZY9I 137661616 IC50 < 10000 nM T20709 C41ZYJ 137701968 EC50 > 30000 nM T20709 C38OTS 145960427 Ki = 177.83 nM T20709 C06LVP 145960466 Ki = 11.48 nM T20709 CSV5D4 145960592 Ki = 165.96 nM T20709 C4KH9G 145960827 Ki = 100 nM T20709 CJI6G2 145961125 Ki = 1174.9 nM T20709 CK7OJ5 145961126 Ki = 2754.23 nM T20709 C0XL7S 145961152 Ki = 8511.38 nM T20709 C3WFT9 145961161 Ki = 22.91 nM T20709 CJ50OV 145961495 Ki = 141.25 nM T20709 CAH97Y 145961981 Ki = 257.04 nM T20709 CH1AE6 145962050 Ki = 512.86 nM T20709 CG16NQ 145963288 Ki = 436.52 nM T20709 CBM12W 145963804 EC50 = 2290 nM T20709 CPQ85Z 145964807 EC50 = 1510 nM T20709 C2Q1TO 145965320 EC50 = 851 nM T20709 CCR58Y 145966183 EC50 = 151 nM T20709 C3LEF7 145966439 EC50 = 15 nM T20709 C0IO4R 145966968 EC50 > 10000 nM T20709 CRP5C4 145968703 EC50 = 457 nM T20709 C52HDU 145970522 EC50 = 1096 nM T20709 CJMR32 145972844 EC50 = 1445.44 nM T20709 CAW4E7 145973064 EC50 = 407 nM T20709 CWQ46M 145973726 EC50 = 57 nM T20709 CMUW76 145974039 EC50 > 10000 nM T20709 CS3YZ7 145976573 EC50 = 324 nM T20709 CU03IC 145976835 EC50 = 331 nM T20709 C5T7ED 145978398 EC50 = 199.53 nM T20709 C5J1DR 145978505 EC50 > 10000 nM T20709 CHIZ91 153284501 IC50 = 12500 nM T20709 C6P3SR 153287553 Ki > 10000 nM T20709 CV9G7Z 153287572 Ki > 10000 nM T20709 CO85KL 153287574 Ki > 10000 nM T20709 CKU28V 155510640 EC50 = 102 nM T20709 CQB01O 155511952 EC50 > 10000 nM T20709 C2BDK6 155513985 Ki = 29.51 nM T20709 C53FKW 155516382 Ki = 23.44 nM T20709 C32DEA 155518224 EC50 = 10000 nM T20709 CB0Y3M 155518790 EC50 = 23 nM T20709 CYO6S2 155519300 EC50 = 20 nM T20709 C6RN8D 155519324 EC50 > 10000 nM T20709 CDV54Q 155519506 EC50 > 10000 nM T20709 C5YDE2 155519621 Ki = 1740 nM T20709 C0MT4Q 155519740 Ki = 6.457 nM T20709 CUSA24 155519891 Ki > 10000 nM T20709 CI7EY8 155520062 EC50 > 10000 nM T20709 C5W7OK 155520162 EC50 = 478.63 nM T20709 C6RD8Y 155520521 EC50 = 3410 nM T20709 CQ5HJ7 155520594 EC50 > 10000 nM T20709 C39OYH 155521109 EC50 = 86 nM T20709 CPVA65 155521382 Ki = 147.91 nM T20709 CFVP27 155521893 Ki = 0.912 nM T20709 CWI7D5 155522181 EC50 = 180 nM T20709 CL9ET5 155522354 Ki = 61.66 nM T20709 C57AIL 155522645 EC50 = 37 nM T20709 CPIL73 155523539 EC50 = 470 nM T20709 CL6O1R 155523647 Ki = 1.072 nM T20709 C38PTA 155523888 Ki = 89.13 nM T20709 C8V5WM 155524827 EC50 = 16 nM T20709 C5P1YE 155525064 Ki = 79.43 nM T20709 CDQ89Y 155525097 Ki = 2.57 nM T20709 CLG04I 155525665 EC50 > 9930 nM T20709 CBK0Y7 155528269 Ki = 257.04 nM T20709 CMD75Z 155529555 EC50 > 8880 nM T20709 CMG17K 155531483 EC50 = 990 nM T20709 C8SM9U 155532238 EC50 = 2510 nM T20709 C7CU8J 155535606 Ki = 2.692 nM T20709 CB79ZW 155536080 Ki > 10000 nM T20709 C6E0PN 155536105 EC50 > 4160 nM T20709 CQBT73 155537519 EC50 > 5990 nM T20709 CW6FY4 155538474 EC50 = 296 nM T20709 C1TKS0 155539410 EC50 = 7 nM T20709 CV1Q2O 155539604 EC50 = 645.65 nM T20709 CV2NG9 155539712 Ki = 3.236 nM T20709 CJRA40 155539719 EC50 = 104.71 nM T20709 CNK15J 155540233 EC50 = 37 nM T20709 CRLS19 155540893 EC50 = 2200 nM T20709 C74WLP 155540988 EC50 > 10000 nM T20709 CE92AJ 155541265 EC50 > 10000 nM T20709 C9OVX7 155541662 EC50 > 10000 nM T20709 CK70MJ 155541812 Ki = 2.2 nM T20709 CK4CP9 155542543 EC50 > 10000 nM T20709 CS5YB1 155543344 Ki = 57.54 nM T20709 COV93Z 155543943 Ki = 3.548 nM T20709 CNIS02 155543990 EC50 = 295 nM T20709 CJ96MW 155544229 EC50 = 588.84 nM T20709 C8ZL6X 155544752 EC50 > 10000 nM T20709 CWHM54 155544761 EC50 > 10000 nM T20709 CQ0MG9 155546031 EC50 = 380 nM T20709 CZ5I7V 155546304 EC50 = 3800 nM T20709 CJXW85 155547285 EC50 = 95 nM T20709 C2CB8H 155548585 Ki = 56.23 nM T20709 C9KBH7 155550435 Ki = 1.122 nM T20709 CRIJ70 155550631 Ki = 2.042 nM T20709 CZ6US1 155550854 EC50 > 10000 nM T20709 CE3F2K 155551015 EC50 = 228 nM T20709 COF49W 155551902 Ki = 208.93 nM T20709 C4D2FT 155552040 EC50 > 10000 nM T20709 CV23QD 155552262 EC50 > 10000 nM T20709 C8LRX2 155552304 EC50 = 9 nM T20709 C7I8XD 155552432 EC50 = 1100 nM T20709 CAB6P1 155552902 EC50 > 10000 nM T20709 CXZQ46 155552922 Ki = 295.12 nM T20709 CAXE16 155553146 EC50 = 76 nM T20709 CBX1Q3 155553357 EC50 > 10000 nM T20709 CB43IP 155554015 EC50 = 331 nM T20709 C7TF1D 155554261 Ki = 93.33 nM T20709 C73DFN 155554567 Ki = 2.455 nM T20709 C0XF4G 155556079 EC50 > 10000 nM T20709 C1TDY8 155556289 Ki = 1.259 nM T20709 C2D3SP 155557118 Ki = 37.15 nM T20709 CT5DG2 155557669 EC50 = 160 nM T20709 CCF1T9 155557847 EC50 > 2740 nM T20709 CJ0CK3 155558680 EC50 > 10000 nM T20709 C75PXS 155559290 Ki = 1071.52 nM T20709 CEAD84 155559740 Ki = 10.72 nM T20709 CO9S4Y 155559816 EC50 > 10000 nM T20709 CP2U8A 155560012 Ki = 27.54 nM T20709 CU3TF1 155560139 Ki = 17.38 nM T20709 CGY0O1 155560153 EC50 = 891 nM T20709 CCO15D 155560304 Ki = 1.202 nM T20709 CJM85L 155561780 EC50 = 3 nM T20709 CF7B0T 155561871 EC50 = 9830 nM T20709 CMX98Q 155562285 Ki = 25 nM T20709 CH9YK4 155562731 EC50 > 10000 nM T20709 CPB8H4 155562860 EC50 = 220 nM T20709 CN4I2Q 155563154 EC50 > 10000 nM T20709 CY21WX 155563393 EC50 = 239.88 nM T20709 C69IUF 155564640 EC50 = 104.71 nM T20709 CVLR58 155565285 Ki = 416.87 nM T20709 CDS7K2 155566289 Ki = 2.089 nM T20709 C83SNF 155566810 EC50 > 10000 nM T20709 CY30EN 155567379 Ki = 1.622 nM T20709 C3DW7M 155569381 EC50 > 9250 nM T20709 C0OB6P 155569594 EC50 > 10000 nM T20709 C3N9VU 10251906 Ki > 500 nM T20709 C9RLJ3 3661 Ki = 0.64 nM T20709 CD6OK3 44455198 Ki = 6.3 nM T20709 D01UDC 9815331 Ki = 4 nM T20709 D02BOW 5926 Ki = 9120.11 nM T20709 D02EXX 3013846 Ki = 140 nM T20709 D02KZD 71598521 IC50 > 30000 nM T20709 D02ZPV 10125445 Ki = 10 nM T20709 D03DKZ 42633508 EC50 > 30000 nM T20709 D03RMI 11536903 Ki = 389.05 nM T20709 D04XNH 44318851 Ki = 85 nM T20709 D05ZUX 44207909 Ki >= 1000 nM T20709 D06IUC 6508730 Ki = 121 nM T20709 D07GPQ 132947 Ki = 6.457 nM T20709 D09RPR 16737207 Ki > 10000 nM T20709 D0A2KT 3014059 Ki = 0.37 nM T20709 D0AR0H 6508724 Ki = 103 nM T20709 D0C2DM 9893054 EC50 = 1060 nM T20709 D0C9ZE 10105296 Ki = 190 nM T20709 D0F5LH 4634 Ki = 3.631 nM T20709 D0FF6S 16038374 IC50 > 10000 nM T20709 D0H4BJ 9308 Ki = 23 nM T20709 D0H8XV 12963076 Ki = 3890.45 nM T20709 D0HP1O 119357 Ki = 10 nM T20709 D0I9LU 2229 Ki = 977.24 nM T20709 D0JV2S 3008304 EC50 > 30000 nM T20709 D0K3HY 864492 EC50 = 520 nM T20709 D0L1XR 4630 Ki = 1.5 nM T20709 D0L5MW 181743 Ki > 10000 nM T20709 D0N2KU 44517677 Ki = 4300 nM T20709 D0P1FJ 71128 Ki = 7.4 nM T20709 D0T2RY 9948320 Ki >= 1000 nM T20709 D0TX8W 594590 Ki > 19952.62 nM T20709 D0WO3A 4141 Ki = 6309.57 nM T20709 D0X7HD 11184481 Ki = 3000 nM T20709 D0Z5RQ 656392 IC50 = 498 nM T20709 D0Z6VT 71737672 EC50 > 30000 nM T10375 D0E3TC 44259 IC50 = 2.33 nM T10375 CACS26 11561968 Ki > 2000 nM T10375 CU0E8O 11690457 Ki > 10000 nM T10375 CLI16E 44465026 IC50 = 3700 nM T10375 CV63UL 67240318 IC50 > 10000 nM T10375 CDP7Q0 134130181 IC50 > 10000 nM T10375 C2MD1Q 155513187 IC50 > 10000 nM T10375 D03BJF 44465558 IC50 = 1900 nM T10375 D0A7FQ 11644425 IC50 = 1100 nM T10375 D0CE3R 5312137 IC50 = 100 nM T21678 D0MU9L 176077 IC50 = 42 nM T21678 D0S5LT 29435 Ki = 18000 nM T21678 C2P0AK 480948 IC50 = 805000 nM T21678 CX76PN 6475030 IC50 = 80000 nM T21678 C90QNU 9882222 IC50 = 9500 nM T21678 CJ6TV8 10011928 IC50 > 1000000 nM T21678 CZT1D2 10080697 Ki = 67000 nM T21678 CE9XP3 10240946 Ki > 2000000 nM T21678 CE2AF4 10352016 IC50 = 920000 nM T21678 CLKA50 11240664 IC50 = 390000 nM T21678 CJE5T9 12103482 IC50 = 14000 nM T21678 CW28RN 12103488 IC50 = 53 nM T21678 CT0JI3 13018788 IC50 = 45000 nM T21678 C40CSF 25181192 IC50 = 22100 nM T21678 CYBM80 44367875 IC50 > 1000000 nM T21678 CF7H4C 44368231 IC50 > 1000000 nM T21678 C75BDZ 44368232 IC50 > 1000000 nM T21678 CS5ZN1 44368239 IC50 = 725000 nM T21678 C1JWV2 46906966 IC50 = 224000 nM T21678 CEP1M9 90664182 Ki = 300000 nM T21678 C9SN4L 90664183 Ki = 400000 nM T21678 CVK90M 102029945 IC50 = 34200 nM T21678 C3WBY2 127025939 Ki > 2000000 nM T21678 C30RWL 127027504 Ki > 2000000 nM T21678 C9J8LD 127027505 Ki > 2000000 nM T21678 C9WSG4 137632720 IC50 = 5000 nM T21678 C2NOP7 137639289 IC50 = 7700 nM T21678 CZJT84 137641705 IC50 = 3000 nM T21678 C4EAZ0 137646452 Ki = 2000 nM T21678 CKFJ47 137656079 IC50 = 13000 nM T21678 C7YNR0 145950365 IC50 = 3500 nM T21678 CDE64Z 145951974 IC50 = 3100 nM T21678 C6M5NI 145956209 IC50 = 1200 nM T21678 C2J4TZ 145956399 Ki = 3500 nM T21678 C2M5WG 145963126 IC50 = 13000 nM T21678 CT0Q8H 145965670 IC50 = 159000 nM T21678 CXZH98 145971016 IC50 = 185000 nM T21678 CE8RL1 145972204 IC50 = 4100 nM T21678 CE40SO 145978797 IC50 = 171000 nM T21678 D07RRH 46906930 IC50 = 15000 nM T21678 D0Q1KL 44320078 IC50 = 6400 nM T21678 D0R8TR 445612 IC50 = 40000 nM T21678 D0RU5N 46906931 IC50 = 39000 nM T21678 D0SQ1T 10261406 Ki = 500 nM T60182 D0H8WF 44278361 EC50 = 0.0004 nM T60182 D0LI1C 44469321 IC50 > 30000 nM T60182 D0V7SO 60151939 Ki = 14 nM T60182 D00NCJ 57388936 Ki = 15 nM T60182 D04NUS 71202253 IC50 = 290 nM T60182 D05AWM 53377591 IC50 = 61 nM T60182 D0AJ3F 53467170 IC50 = 22 nM T60182 D0F9RK 53377590 IC50 = 209 nM T60182 D0IT9C 71472272 Ki = 17 nM T60182 D0JA0A 68178614 Ki = 690 nM T60182 D00MEV 160115 IC50 = 20000 nM T60182 D0F8DL 176155 IC50 = 37.07 nM T60182 D0Z6AX 5311277 Ki = 356 nM T60182 CK0JH3 416615 Ki > 500000 nM T60182 CAN65C 654283 Ki = 55000 nM T60182 C1KQ2D 677928 Ki > 60000 nM T60182 CZN6S9 743974 EC50 > 50118.72 nM T60182 C8B5NS 747420 Ki > 500000 nM T60182 CP5L9K 825433 Ki > 500000 nM T60182 CV0Q3D 1302369 IC50 > 30000 nM T60182 C0GE2X 1619763 IC50 > 30000 nM T60182 CE9Q7X 1714260 IC50 = 2200 nM T60182 C21HKV 1941609 IC50 > 30000 nM T60182 CQ48HM 2228665 Ki = 42000 nM T60182 C8I9FA 3652254 IC50 = 870 nM T60182 CJ8X2U 4047161 IC50 > 20000 nM T60182 CDG5X2 4066568 Ki = 73000 nM T60182 COSL39 4450383 Ki = 250000 nM T60182 CWHE97 6862006 IC50 = 1800 nM T60182 CG5TP3 6875509 IC50 = 4900 nM T60182 C08UWD 9555433 IC50 = 4800 nM T60182 CE0YO6 9824797 IC50 = 84 nM T60182 CJ7T9X 9825482 IC50 = 5.3 nM T60182 C6GSZ2 9836535 IC50 = 130.02 nM T60182 C83VNA 9841863 IC50 = 490 nM T60182 C1EX9P 9843239 IC50 = 130 nM T60182 C68YGH 9869430 IC50 = 27.5 nM T60182 CS02XG 9871912 IC50 = 130 nM T60182 CXJ85S 9873139 IC50 = 631 nM T60182 CJ4QV2 9885993 IC50 = 5.309 nM T60182 CU5O0E 9886904 IC50 = 90.16 nM T60182 C57EYC 9891138 IC50 = 6.5 nM T60182 CS7HU2 9902041 IC50 = 2000 nM T60182 C7H2LE 9906120 IC50 = 110 nM T60182 CF6AV4 9914410 IC50 = 166 nM T60182 CP96LK 9916972 IC50 = 9 nM T60182 CF69AC 9929037 IC50 = 810 nM T60182 C3BPW2 9938390 Ki = 4 nM T60182 CU0Z3A 9946911 IC50 = 50 nM T60182 C8OI3N 9952509 IC50 = 160.03 nM T60182 C1UX9C 9955419 IC50 = 2.3 nM T60182 CUCW87 9956429 IC50 = 33.8 nM T60182 CNW2J4 9957123 IC50 = 22.9 nM T60182 C8B7LA 9983854 IC50 = 2900 nM T60182 CHSN85 9985258 IC50 = 93 nM T60182 CGEJ24 9985625 IC50 = 113.8 nM T60182 CV0QE1 9986018 IC50 = 92 nM T60182 CUG3X7 9998923 IC50 = 1500 nM T60182 CP7H1R 10007881 IC50 = 36 nM T60182 CKEO50 10007966 IC50 = 43 nM T60182 CC24LY 10008376 IC50 = 95 nM T60182 CQ3ED0 10008709 IC50 = 1965 nM T60182 CF86IP 10030697 IC50 = 76 nM T60182 CRU48M 10030948 IC50 = 480 nM T60182 C6LHS9 10031040 IC50 = 336 nM T60182 C6L7UO 10032265 IC50 = 3.9 nM T60182 C1U5SW 10044081 IC50 = 3210 nM T60182 C6E9ZH 10052441 IC50 = 94 nM T60182 COC68H 10053841 IC50 = 35 nM T60182 CVMB14 10053876 IC50 = 4.6 nM T60182 CXFW65 10053886 IC50 = 53 nM T60182 CR6NW9 10054055 IC50 = 32 nM T60182 C7Q9XL 10054432 IC50 = 7200 nM T60182 C01SHG 10066912 IC50 = 280.54 nM T60182 C7THV5 10072624 IC50 = 2556 nM T60182 C5D3QP 10073298 IC50 = 1663 nM T60182 CKW04V 10073574 IC50 = 20 nM T60182 CT08NW 10076778 IC50 = 2400 nM T60182 CLQM81 10076914 IC50 = 560 nM T60182 CH0ZK9 10076995 IC50 = 220 nM T60182 CZXK14 10077065 IC50 = 2700 nM T60182 C1BKD9 10077102 IC50 = 856 nM T60182 C4P6KU 10077369 IC50 = 130 nM T60182 CNZS08 10093802 IC50 = 6.5 nM T60182 CK05GO 10097880 IC50 = 810 nM T60182 CC1UA3 10099927 IC50 = 282 nM T60182 CY6E8O 10133915 IC50 = 300.61 nM T60182 C0P5DE 10144347 IC50 = 9 nM T60182 C0B5WP 10144633 IC50 = 18 nM T60182 C62RYU 10144925 IC50 = 51 nM T60182 CFD96W 10145290 IC50 = 693 nM T60182 C70HKJ 10145603 IC50 = 14 nM T60182 CTR46Q 10167904 IC50 = 6 nM T60182 C85IFN 10168348 IC50 = 6 nM T60182 C6CH8L 10210150 IC50 = 55 nM T60182 CQ0NT1 10211765 IC50 = 7 nM T60182 C4S9MD 10211943 IC50 = 5 nM T60182 CGAP51 10215420 IC50 = 100 nM T60182 C0B2DH 10231964 IC50 = 14 nM T60182 C8CNK1 10232009 IC50 = 4 nM T60182 C2LM1T 10246001 IC50 = 90.16 nM T60182 C8R7YJ 10255803 IC50 = 16000 nM T60182 C08BCM 10257357 IC50 = 12 nM T60182 C4ZA2X 10257529 IC50 = 60 nM T60182 CDZ62K 10257629 IC50 = 54 nM T60182 CQ49SX 10280734 IC50 = 14 nM T60182 CMW97S 10282059 IC50 = 8 nM T60182 CW16YI 10282162 IC50 = 13 nM T60182 C09YQC 10282370 IC50 = 9 nM T60182 CL19HJ 10318451 IC50 = 150.31 nM T60182 CA10KJ 10323446 IC50 = 700 nM T60182 CMK7Q6 10324097 IC50 = 120 nM T60182 C4RET3 10324098 IC50 = 4200 nM T60182 CVA4W8 10325599 IC50 = 407 nM T60182 CH20FQ 10326056 IC50 = 43 nM T60182 CS7NA4 10338890 IC50 = 23.01 nM T60182 CTHC17 10346647 IC50 = 116 nM T60182 C2T4HR 10360917 Ki = 5400 nM T60182 C69ZYI 10363819 IC50 = 8.5 nM T60182 CI4G2Z 10369244 IC50 = 7200 nM T60182 CO5PW3 10369510 IC50 = 27 nM T60182 CB56SY 10369580 IC50 = 601 nM T60182 CPVK45 10370821 IC50 = 105 nM T60182 CHG60B 10383925 IC50 = 185 nM T60182 CL5RY9 10393857 IC50 = 1691 nM T60182 C1V8EH 10393937 IC50 = 51 nM T60182 C6Z1HO 10413333 IC50 = 59 nM T60182 CRCP21 10415723 IC50 = 39 nM T60182 C1H7ZQ 10415955 IC50 = 1200 nM T60182 C04QSL 10416067 IC50 = 30 nM T60182 CY7S9E 10416258 IC50 = 1100 nM T60182 CUHG87 10434112 IC50 = 11.6 nM T60182 CPBQ83 10435275 IC50 = 41 nM T60182 CG4DC1 10435562 IC50 = 894 nM T60182 C0BJQ4 10436553 IC50 = 3800 nM T60182 C68PTF 10436554 IC50 = 1700 nM T60182 C9EXA7 10437700 IC50 = 1416 nM T60182 C0ULD9 10438267 IC50 = 570 nM T60182 C4O1JU 10450820 IC50 = 870 nM T60182 CIRO42 10459436 IC50 = 65 nM T60182 CC1FQ2 10461010 IC50 = 120 nM T60182 CO87CR 10461326 IC50 = 250 nM T60182 C8H1AN 10474631 IC50 = 40.09 nM T60182 CK4A7P 10481623 IC50 = 2900 nM T60182 CAR05Z 10481840 IC50 = 739 nM T60182 CF8I6B 10483282 IC50 = 10 nM T60182 CF7YP9 10483611 IC50 = 370 nM T60182 CW1PQ2 10519171 Ki > 500000 nM T60182 CF87WH 10552082 Ki = 16000 nM T60182 CXH3D5 10592750 IC50 = 2000 nM T60182 CM56AS 10600858 Ki = 9200 nM T60182 CC14YF 10613052 Ki = 380000 nM T60182 CP51TX 10617488 Ki = 55000 nM T60182 CF7K2X 10638990 Ki > 500000 nM T60182 CM16SH 10640008 Ki > 500000 nM T60182 CB94VU 10686727 Ki = 41000 nM T60182 CW8FL5 10687711 Ki = 200000 nM T60182 C5TB2X 10692484 Ki = 180000 nM T60182 CD4EI0 10694841 Ki = 95000 nM T60182 CB0M7J 10716305 Ki = 18000 nM T60182 C90TEL 10729333 Ki > 500000 nM T60182 CWQ2E9 10757473 Ki > 500000 nM T60182 C7PQM1 10804979 Ki = 160000 nM T60182 CO70NH 10829406 Ki = 12000 nM T60182 CG92SJ 10829563 Ki > 500000 nM T60182 CYMC13 10854791 Ki > 500000 nM T60182 CI45ZW 10864173 IC50 = 13.8 nM T60182 CE0GN3 10864579 IC50 = 4.9 nM T60182 C0WAU7 10864629 IC50 = 54.3 nM T60182 C8JX1D 10873618 IC50 = 2540 nM T60182 C1M4WD 10882636 IC50 = 2900 nM T60182 C9UCN3 10907299 IC50 = 5.9 nM T60182 C5LN4C 10907780 IC50 = 14.5 nM T60182 C1HQ0K 10918616 IC50 = 7.9 nM T60182 CDNC71 10924293 IC50 > 100000 nM T60182 CYH8Z7 10928006 IC50 = 33 nM T60182 CES92X 10929597 IC50 = 9.2 nM T60182 C1MVP3 10951675 IC50 = 14.7 nM T60182 CF53ON 10951864 IC50 = 11.3 nM T60182 C2HT7B 10957546 IC50 > 100000 nM T60182 CXT18Z 10960967 IC50 = 4900 nM T60182 CRD87T 10962252 IC50 = 51.7 nM T60182 CPQ3M5 10962393 IC50 = 133 nM T60182 C4AZ3F 10970292 IC50 = 41.1 nM T60182 CJH26P 10971714 IC50 = 6.4 nM T60182 CN06LB 10973527 IC50 = 73 nM T60182 CPBR67 10974243 IC50 = 11.4 nM T60182 CBC87Z 10980170 IC50 = 10000 nM T60182 CTB3M0 10981564 IC50 > 100000 nM T60182 CH92PV 10982999 IC50 = 22.6 nM T60182 CI8XA0 10992755 IC50 = 53.8 nM T60182 C2A0TR 10995358 IC50 = 19.7 nM T60182 C29EKI 11001603 IC50 > 100000 nM T60182 CG3F4B 11003592 IC50 = 6300 nM T60182 C9K0EX 11024220 IC50 = 29.4 nM T60182 CKJ29N 11024350 IC50 = 120.23 nM T60182 C4YZH9 11027864 IC50 = 10.4 nM T60182 C9EH6R 11034750 IC50 = 29000 nM T60182 C2DJB6 11037917 IC50 = 28.7 nM T60182 C9NCS2 11038653 IC50 = 2.8 nM T60182 CSBM25 11039347 IC50 = 6.1 nM T60182 CR7KP2 11045195 IC50 = 43000 nM T60182 CST41Y 11045899 IC50 > 100000 nM T60182 CB0X1M 11048133 IC50 = 35.4 nM T60182 C6CDH5 11048232 IC50 = 16.5 nM T60182 C5U9NG 11048896 IC50 = 268 nM T60182 CKAP89 11049295 IC50 = 90.6 nM T60182 CN53YG 11049977 IC50 = 27.7 nM T60182 C3L7ZB 11057703 IC50 = 75.5 nM T60182 C3HX8W 11068219 IC50 = 200 nM T60182 C7Z0PA 11068479 IC50 = 8100 nM T60182 C12MOG 11078726 IC50 = 43000 nM T60182 C2RJ1P 11081564 IC50 = 47.8 nM T60182 CD51TR 11082135 IC50 = 12.3 nM T60182 CRSW28 11091831 IC50 = 8.3 nM T60182 C20PMB 11102152 IC50 = 38.8 nM T60182 C9NEK5 11102344 IC50 = 5.8 nM T60182 C1UQO0 11102467 IC50 = 49.7 nM T60182 CFX2D4 11103530 IC50 = 6.2 nM T60182 CF07SG 11113396 IC50 = 441 nM T60182 CGP8K2 11113699 IC50 = 286 nM T60182 CDIV09 11114038 IC50 = 33.5 nM T60182 CXBJ59 11142525 IC50 = 26000 nM T60182 CBU42D 11145271 IC50 = 120 nM T60182 CSC62V 11145871 IC50 = 3.4 nM T60182 CP4E5W 11157621 IC50 = 18 nM T60182 C41AIU 11169089 IC50 = 1 nM T60182 CZQ7W3 11180162 IC50 = 80 nM T60182 C13COS 11186974 IC50 = 220 nM T60182 C4R2NX 11238073 IC50 = 18 nM T60182 CPN60U 11238149 IC50 = 950 nM T60182 CG8B7V 11238814 IC50 = 64 nM T60182 CU4J6H 11249762 IC50 = 2 nM T60182 C7W1XE 11250000 IC50 = 55 nM T60182 CHL1X3 11260553 IC50 = 16 nM T60182 CP7B1L 11261540 IC50 = 16 nM T60182 CRCL23 11273570 IC50 = 14.4 nM T60182 CHR6C3 11283703 IC50 = 24 nM T60182 CG29RY 11284556 IC50 = 12 nM T60182 C4H3RQ 11284982 IC50 = 7 nM T60182 C5XMJ8 11308245 IC50 = 3.1 nM T60182 C2TIO4 11329242 IC50 = 10 nM T60182 CO2CQ7 11331120 IC50 = 1.3 nM T60182 C03EMK 11352330 IC50 = 230 nM T60182 C68VWR 11352703 IC50 = 90 nM T60182 COE04Q 11352811 IC50 = 18 nM T60182 CPQ15F 11353908 IC50 = 9.3 nM T60182 CP1VF4 11365464 IC50 = 11 nM T60182 CG43XJ 11376210 IC50 = 1 nM T60182 COG94K 11383934 IC50 = 20000 nM T60182 CJX58D 11387112 IC50 = 110 nM T60182 CGP2D8 11410772 IC50 = 24 nM T60182 C8J4UT 11410779 IC50 = 1 nM T60182 CGY9X6 11421820 IC50 = 4.4 nM T60182 C7R8ZB 11421826 IC50 = 4 nM T60182 CNLC72 11432140 IC50 = 28 nM T60182 CFYK03 11433550 IC50 = 640 nM T60182 CC5WD2 11444850 IC50 = 2.2 nM T60182 CE16VH 11456034 IC50 = 13 nM T60182 CJ4K2U 11456187 IC50 = 8.3 nM T60182 C3MQO9 11478813 IC50 = 7 nM T60182 C49IQP 11490222 IC50 = 30 nM T60182 COE89G 11490393 IC50 = 8.3 nM T60182 C4YR5H 11527170 IC50 = 298 nM T60182 C0N6UB 11527207 IC50 = 7.5 nM T60182 CR4M7L 11559533 IC50 = 17000 nM T60182 CB59HM 11570626 IC50 = 6.6 nM T60182 CR78YS 11585375 IC50 = 10.7 nM T60182 C3JE1T 11585452 IC50 = 16.6 nM T60182 C1BT6K 11592461 IC50 = 8.1 nM T60182 CP56DO 11599295 IC50 = 11 nM T60182 CCQZ38 11621378 IC50 = 12.3 nM T60182 C5J9XZ 11650288 IC50 = 121.5 nM T60182 CW8LD3 11657413 IC50 = 8.1 nM T60182 C7RI5K 11678966 IC50 = 64.2 nM T60182 CLY98H 11678967 IC50 = 40.5 nM T60182 C4B2JQ 11699553 IC50 = 58.5 nM T60182 CN7RJ8 11731304 IC50 = 96.7 nM T60182 CITQ01 11733947 IC50 = 15.7 nM T60182 CJ8M0A 11754125 IC50 = 89 nM T60182 C3RZF0 11756248 IC50 = 1200 nM T60182 C8FC6B 11757662 IC50 = 156 nM T60182 CU56HZ 11757679 IC50 = 63 nM T60182 C7Y5JE 11760806 IC50 = 12000 nM T60182 CE0CZ6 11764614 IC50 = 82 nM T60182 CSZQ52 11764615 IC50 = 8 nM T60182 CL03NR 11782911 IC50 = 29.8 nM T60182 C5MUB1 11785044 IC50 = 4 nM T60182 C1QV9Z 11786041 IC50 = 120 nM T60182 C5ES4P 11793430 Ki = 20000 nM T60182 C3KHU4 11809785 IC50 > 100000 nM T60182 CD71PU 11812426 IC50 = 19.1 nM T60182 C17GTD 11813262 IC50 = 485 nM T60182 CYH3V9 11814151 IC50 = 6.6 nM T60182 CQ6C2O 11826682 IC50 = 22.3 nM T60182 C56OQC 11826907 IC50 = 7.4 nM T60182 C4XEG6 11827809 IC50 = 89.3 nM T60182 CK25CM 11949739 IC50 = 28 nM T60182 CTM6N5 11949740 IC50 = 7.6 nM T60182 CNI85P 11950075 IC50 = 500 nM T60182 CL2GD7 11950794 IC50 = 1052 nM T60182 CSV4A0 11950795 IC50 = 54 nM T60182 C6BYQ0 11950971 IC50 = 4.8 nM T60182 CM2XR7 11950972 IC50 = 39 nM T60182 CMKB05 11951681 IC50 = 68 nM T60182 CK6I9N 11951857 IC50 = 22 nM T60182 C7H2SG 11952035 IC50 = 15 nM T60182 CQ0KU7 11952211 IC50 = 33 nM T60182 C1SJ5W 11952213 IC50 = 49 nM T60182 C3A7CL 11952214 IC50 = 4.8 nM T60182 C7VI6D 11952394 IC50 = 4.9 nM T60182 C0XE2H 12967031 IC50 = 800 nM T60182 C7N4DA 12967032 IC50 = 40 nM T60182 CAVB53 12967033 IC50 = 420.73 nM T60182 CR91OX 12967034 IC50 = 80.17 nM T60182 C86PGJ 12967035 IC50 = 260 nM T60182 CHOU39 15407872 IC50 = 210.38 nM T60182 C61OFZ 15924226 IC50 > 20000 nM T60182 COF34S 16100296 IC50 = 21 nM T60182 CKX87Y 16100297 IC50 = 1045 nM T60182 C5JXN1 16100298 IC50 = 226 nM T60182 CMQX07 16100299 IC50 = 35 nM T60182 C05PIH 16100300 IC50 = 16 nM T60182 C3IKW1 16100301 IC50 = 2429 nM T60182 CI40VG 16100302 IC50 = 140 nM T60182 C8RF9J 16100303 IC50 = 215 nM T60182 CM3YF6 16100304 IC50 = 153 nM T60182 CI7X1N 16100305 IC50 = 182 nM T60182 C8Y9RM 16100306 IC50 = 80 nM T60182 CK1PO9 16100307 IC50 > 10000 nM T60182 CG45PD 16100308 IC50 > 10000 nM T60182 CF03KX 16100309 IC50 > 10000 nM T60182 CI89VJ 16100310 IC50 = 1984 nM T60182 C30TKC 16100311 IC50 = 122 nM T60182 CV02TW 16100312 IC50 = 1207 nM T60182 CE38YS 16100313 IC50 = 137 nM T60182 CJ8T3R 16100314 IC50 = 167 nM T60182 CI4AL2 16100315 IC50 = 262 nM T60182 C02WZT 16100316 IC50 = 61 nM T60182 CD7R9P 16100318 IC50 > 10000 nM T60182 C3NO2B 16100319 IC50 = 1700 nM T60182 CVW0U8 16100320 IC50 > 10000 nM T60182 C95ZXG 16100321 IC50 = 2960 nM T60182 C2I0YP 16100327 IC50 = 1088 nM T60182 C9Y0ZP 16100330 IC50 > 10000 nM T60182 CT97KI 16100331 IC50 = 782 nM T60182 CF8W5R 16100332 IC50 = 59 nM T60182 CE04TC 16100333 IC50 = 528 nM T60182 C53GHR 16100334 IC50 = 96 nM T60182 C8E5AQ 16100335 IC50 = 571 nM T60182 CW5DM8 16100336 IC50 = 179 nM T60182 CB27HR 16100337 IC50 > 10000 nM T60182 C9R4NO 16100338 IC50 = 1000 nM T60182 C0XP5O 16100339 IC50 > 10000 nM T60182 C3IL9B 16199250 EC50 = 1.68 nM T60182 CWG93N 16223791 IC50 = 23 nM T60182 CNF1S6 16223987 IC50 = 28 nM T60182 CXV6I8 16224190 IC50 = 120 nM T60182 CB3UD6 16224191 IC50 = 58 nM T60182 CS6AF1 16224591 IC50 = 24 nM T60182 CL9ZC8 16224781 IC50 = 28 nM T60182 C0E2WI 16225177 IC50 = 110 nM T60182 C8Y3EI 16225178 IC50 = 16 nM T60182 C0VB6O 16225179 IC50 = 12 nM T60182 CH0SU2 16225393 IC50 = 47 nM T60182 CKF31S 16225394 IC50 = 32 nM T60182 C7CGX6 18926938 IC50 = 9000 nM T60182 CU96LD 19072340 IC50 = 1100 nM T60182 C02SWO 19072347 IC50 = 190.11 nM T60182 CYF76O 20647512 IC50 = 11000 nM T60182 C8EW9L 20674619 IC50 = 521.19 nM T60182 CR06WQ 20742348 Ki = 51 nM T60182 CGC2I1 20775791 IC50 = 225 nM T60182 CB7ID8 20775792 IC50 = 261 nM T60182 C29FRA 20775916 IC50 = 99 nM T60182 C97VQA 20776096 IC50 = 81 nM T60182 CSH17F 20776097 IC50 = 78 nM T60182 C5CE3S 21704177 IC50 = 931.11 nM T60182 C0R9AV 22004872 IC50 = 300 nM T60182 CFR8H4 22004877 IC50 = 1000 nM T60182 CXOK81 22004897 IC50 = 6000 nM T60182 CB8RI4 22004908 IC50 = 9500 nM T60182 C64NCR 22004918 IC50 = 1000 nM T60182 C1FZS0 22004948 IC50 = 19000 nM T60182 CGZ61T 22004955 IC50 = 400 nM T60182 C15ORT 22004988 IC50 = 240 nM T60182 CF05HA 22005015 IC50 = 350 nM T60182 CJQ05X 22005048 IC50 = 48000 nM T60182 C0NM3R 22005050 IC50 = 9000 nM T60182 C2GWD5 22005069 IC50 = 700 nM T60182 CSEK89 22005107 IC50 = 750 nM T60182 CQN08Y 22005108 IC50 > 20000 nM T60182 C94IJS 22005111 IC50 = 1800 nM T60182 CW8H6N 22005118 IC50 = 1800 nM T60182 CPU40C 22005133 IC50 = 6000 nM T60182 CPXL87 22005204 IC50 = 400 nM T60182 CM40EZ 22005216 IC50 > 20000 nM T60182 C9W8GQ 22005250 IC50 = 250 nM T60182 CC5ED0 22005273 IC50 = 7500 nM T60182 C90IJX 22005295 IC50 = 20000 nM T60182 CO2W8L 22005335 IC50 = 1400 nM T60182 CF42TM 22005339 IC50 = 1000 nM T60182 C02USO 22005341 IC50 = 1100 nM T60182 C0MNO2 22005361 IC50 = 800 nM T60182 C5UY8B 22005388 IC50 = 3000 nM T60182 CK91GP 22496358 IC50 = 153 nM T60182 CQ42EI 22496365 IC50 = 36 nM T60182 CMVS81 22496371 IC50 = 48 nM T60182 C4KL3V 22496373 IC50 = 531 nM T60182 CKXG15 22496384 IC50 = 38 nM T60182 C1YAO5 22496395 IC50 = 315 nM T60182 CG45BT 22496412 IC50 = 118 nM T60182 C86YBZ 22496431 IC50 = 86 nM T60182 CPRG93 22496441 IC50 = 420 nM T60182 CZR6D0 22496445 IC50 = 85 nM T60182 CFE72V 22496448 IC50 = 98 nM T60182 C7NZ5H 22496449 IC50 = 50 nM T60182 CRI13U 22496451 IC50 = 34 nM T60182 CCI62H 22496457 IC50 = 34 nM T60182 C49VUW 22496459 IC50 = 64 nM T60182 CK78ZG 22496477 IC50 = 48 nM T60182 CSV48P 22496546 IC50 = 131 nM T60182 CE8UB0 22496557 IC50 = 93 nM T60182 CHS9Y2 22999282 IC50 = 1200 nM T60182 C7JW4V 23550062 IC50 = 46 nM T60182 C03JNO 42617999 IC50 = 119 nM T60182 C3F2XB 44275043 IC50 = 2300 nM T60182 C1Z3YB 44275085 IC50 = 7000 nM T60182 CQUB12 44304524 Ki = 11 nM T60182 CSG47O 44304525 Ki = 80 nM T60182 CJCT80 44304570 Ki = 26 nM T60182 CVG1W6 44304581 Ki = 73 nM T60182 C3ET1U 44304582 Ki = 70 nM T60182 CCR41L 44304622 Ki = 6 nM T60182 CQ6Z2N 44304623 Ki = 400 nM T60182 CM5EP0 44304770 Ki = 6 nM T60182 C2V6RG 44304771 Ki = 29 nM T60182 C4D7PC 44304787 Ki = 26 nM T60182 CMQY30 44304788 Ki = 66 nM T60182 CT5Z3Y 44304825 Ki = 9 nM T60182 C6ZB8E 44304828 Ki > 5000 nM T60182 CX3VC2 44304835 Ki = 6 nM T60182 C6UT0A 44304913 Ki = 5000 nM T60182 C1I0RU 44304965 Ki = 11 nM T60182 CTH50C 44304982 Ki = 112 nM T60182 CLB1S3 44304993 Ki = 3 nM T60182 C72WKX 44318934 IC50 = 150 nM T60182 CJN1G9 44318935 IC50 = 3303.7 nM T60182 CF13QV 44318950 IC50 = 130 nM T60182 CN7V6L 44318988 IC50 = 2200 nM T60182 CRST01 44319245 IC50 = 100 nM T60182 C8N1GE 44319257 IC50 = 50 nM T60182 C9F0GZ 44319258 IC50 = 20.04 nM T60182 C5I2EM 44319276 IC50 = 300.61 nM T60182 CW2RD6 44319442 IC50 = 190.11 nM T60182 C7R2WM 44319474 IC50 = 27 nM T60182 CGJ5Q1 44319495 IC50 = 13 nM T60182 CW5UT8 44319496 IC50 = 61 nM T60182 C0T7JQ 44319591 IC50 = 400 nM T60182 CV2OF7 44319617 IC50 = 100 nM T60182 C0RC6E 44319681 IC50 = 860.99 nM T60182 CQJ9K8 44319712 IC50 = 2800 nM T60182 CQP80V 44319713 IC50 = 13 nM T60182 CTCE98 44324149 IC50 = 44.06 nM T60182 CW2CV1 44342725 IC50 = 2000 nM T60182 CVO8E1 44361158 IC50 = 150 nM T60182 CINP74 44361161 IC50 > 20000 nM T60182 CK1AI4 44361298 IC50 = 120 nM T60182 C1N9YS 44368911 IC50 = 4.3 nM T60182 C3RA5C 44369018 IC50 = 357 nM T60182 CYJ05Z 44369073 IC50 = 58 nM T60182 C2XA5Y 44369092 IC50 = 8.3 nM T60182 CQ7SJ2 44369100 IC50 = 63.2 nM T60182 CZEB53 44369291 IC50 = 305 nM T60182 C9VEO5 44369318 IC50 = 181 nM T60182 CWN3G2 44369346 IC50 = 615 nM T60182 CIMO40 44372376 IC50 = 90.16 nM T60182 CAD1P9 44372396 IC50 = 320.63 nM T60182 CZ6T1E 44372397 IC50 = 140 nM T60182 CT8K9G 44372405 IC50 = 801.68 nM T60182 CRP9D1 44372406 IC50 = 180.3 nM T60182 CC6NH7 44372451 IC50 > 3000 nM T60182 CE5TI8 44372454 IC50 = 90 nM T60182 C1R5IV 44372471 IC50 = 6 nM T60182 C6VFJ4 44372477 IC50 = 100 nM T60182 CE72TG 44372478 IC50 = 3032 nM T60182 C4QMX9 44372556 IC50 = 290 nM T60182 CPZJ67 44372577 IC50 = 160.32 nM T60182 CXN20W 44372638 IC50 = 90 nM T60182 CW9A4U 44372650 IC50 = 590 nM T60182 CO54NJ 44372661 IC50 > 3000 nM T60182 CA83ZQ 44372671 IC50 = 60 nM T60182 CU08DK 44372676 IC50 = 500 nM T60182 CJ42WU 44372677 IC50 = 70 nM T60182 CYNM09 44372688 IC50 = 8 nM T60182 C0I9AX 44372700 IC50 = 26 nM T60182 C36GFB 44372701 IC50 = 140 nM T60182 C0L8YS 44372720 IC50 = 100 nM T60182 C3LP6U 44372846 IC50 = 1361.44 nM T60182 C7X0JK 44372847 IC50 = 1690.44 nM T60182 C14DKZ 44372856 IC50 = 850 nM T60182 CZPE27 44372870 IC50 = 4 nM T60182 CFOC83 44372888 IC50 = 210.38 nM T60182 C6R7OP 44372904 IC50 = 30 nM T60182 CU6O1J 44372923 IC50 = 40 nM T60182 CPKI70 44372946 IC50 = 60 nM T60182 CFL6I9 44372948 IC50 = 10 nM T60182 CER69Z 44373083 IC50 = 50 nM T60182 C0CBK8 44373103 IC50 = 260.02 nM T60182 C0DSU1 44373191 IC50 = 40 nM T60182 CFEW63 44373192 IC50 = 3 nM T60182 C5A4YX 44373213 IC50 = 20 nM T60182 CVO60Z 44373462 IC50 = 390 nM T60182 C2K9GN 44373463 IC50 = 740 nM T60182 CW40DX 44373464 IC50 = 30000 nM T60182 CB1FE2 44373486 IC50 = 31 nM T60182 CS3UB6 44373502 IC50 = 690 nM T60182 COKY62 44373520 IC50 > 100000 nM T60182 C9LP8M 44373527 IC50 = 50 nM T60182 CNSI58 44373547 IC50 = 110 nM T60182 CP3F0X 44373553 IC50 = 1500 nM T60182 C1VW7B 44373554 IC50 = 940 nM T60182 C4QHO1 44373564 IC50 = 78300 nM T60182 C80TGN 44373585 IC50 = 2700 nM T60182 CBI0Z4 44373586 IC50 = 330 nM T60182 CP12UQ 44373635 IC50 = 1300 nM T60182 CT27OI 44373649 IC50 = 6400 nM T60182 CK56VN 44373676 IC50 = 180 nM T60182 C32BCF 44373707 IC50 = 1900 nM T60182 C5QU8B 44373708 IC50 = 880 nM T60182 CTB97G 44373730 IC50 = 48 nM T60182 C30HJN 44373781 IC50 = 150 nM T60182 CVD12P 44373782 IC50 = 23 nM T60182 C8GUF7 44373783 IC50 = 140 nM T60182 CA5LZ6 44373923 IC50 = 160 nM T60182 CHPI49 44373924 IC50 = 690 nM T60182 CM5U4J 44389584 IC50 = 3820 nM T60182 C98QFV 44389598 IC50 = 59 nM T60182 CQG7P6 44389632 IC50 = 63 nM T60182 CEV1F7 44404222 IC50 = 178 nM T60182 CI7J5B 44404227 IC50 = 113 nM T60182 CW4BL2 44404234 IC50 = 427 nM T60182 C4T5MJ 44404243 IC50 = 33 nM T60182 C0S3MP 44411059 IC50 = 55000 nM T60182 C7C5PE 44411371 IC50 = 35000 nM T60182 CP73KL 44418927 IC50 = 56 nM T60182 CYI26V 44418928 IC50 = 141 nM T60182 C45SUE 44418929 IC50 = 116 nM T60182 C2A1UO 44418950 IC50 = 7000 nM T60182 COCX59 44431011 IC50 = 820 nM T60182 C2IWY5 44431012 IC50 = 3434 nM T60182 CNHM07 44431016 IC50 = 130 nM T60182 C8HOD7 44431020 IC50 = 11 nM T60182 CJ1IL4 44561285 IC50 = 482 nM T60182 CYDE03 44561286 IC50 > 1000 nM T60182 CZ1M7Q 44561287 IC50 = 85 nM T60182 C0IDG4 44561327 IC50 = 15 nM T60182 CW9F1X 44561359 IC50 > 1000 nM T60182 C6I7OF 44561390 IC50 = 31 nM T60182 C5B9GH 44561391 IC50 = 2 nM T60182 C6F4EX 44561438 IC50 = 4 nM T60182 CSB74O 44561439 IC50 = 2 nM T60182 C5A8MI 44561440 IC50 = 19 nM T60182 CQU45G 44561479 IC50 = 4 nM T60182 CE4N0X 44561480 IC50 = 6 nM T60182 CXI09W 44561519 IC50 = 7 nM T60182 C9Y2NP 44561556 IC50 = 9 nM T60182 CCRV56 44561557 IC50 = 160 nM T60182 C9D8EI 44561584 IC50 = 14 nM T60182 CYAI96 44575544 IC50 = 4 nM T60182 CLCK02 44584363 IC50 = 320 nM T60182 C5OPK9 45381049 IC50 = 38 nM T60182 CN0PU9 45381051 IC50 = 380 nM T60182 CS5XO8 45381153 IC50 = 72 nM T60182 CD2VE9 45381268 IC50 = 2200 nM T60182 C0RIG3 45381379 IC50 = 22 nM T60182 C8UY2B 45381380 IC50 = 15 nM T60182 CH13AF 45381381 IC50 = 370 nM T60182 CQS1U6 45485585 EC50 > 10000 nM T60182 CJ16QC 46240797 Ki = 4 nM T60182 CD48CL 49864564 EC50 = 0.47 nM T60182 C37MEV 49864565 EC50 = 0.068 nM T60182 CE9NY7 49864573 EC50 = 2.4 nM T60182 CWKH42 49864580 EC50 = 0.59 nM T60182 C1SG5P 49864615 EC50 = 0.055 nM T60182 CS3Y7O 51031037 IC50 = 130 nM T60182 C6RE3Z 53316573 IC50 = 330 nM T60182 C0OFJ6 53319214 IC50 = 1100 nM T60182 CHRM05 53320525 IC50 = 520 nM T60182 CB2AN5 53321835 IC50 = 1100 nM T60182 CJ46YT 53323150 IC50 = 430 nM T60182 CFTG29 53323247 IC50 = 2000 nM T60182 CH4N5O 53324505 IC50 = 730 nM T60182 CFU20M 53325823 IC50 = 5300 nM T60182 CG2M3A 53325824 IC50 = 28 nM T60182 C2U7FZ 53325825 IC50 = 2900 nM T60182 CRT2V5 53466721 IC50 = 4500 nM T60182 CO3KV0 53466723 IC50 = 8500 nM T60182 CZ9MH8 53469056 IC50 = 44 nM T60182 CS0P9Y 53469058 IC50 = 260 nM T60182 CN3O7H 53469258 IC50 = 510 nM T60182 CD2X1W 53469443 IC50 = 24 nM T60182 CU4R6T 53469628 IC50 = 48 nM T60182 CU09OX 53469820 IC50 = 2700 nM T60182 CL7O5U 53469821 IC50 = 270 nM T60182 C6TEK8 54765284 IC50 = 6 nM T60182 C0T3KY 54765285 IC50 = 12 nM T60182 C97STZ 56602804 IC50 = 3700 nM T60182 C7C9FR 57388856 Ki = 22 nM T60182 CS5Y8C 57390853 IC50 = 450 nM T60182 CHK49F 57390854 IC50 = 37 nM T60182 CH8P3M 57391489 IC50 = 18 nM T60182 C6FVD3 57391519 IC50 = 13 nM T60182 CG48UI 57391683 Ki = 214 nM T60182 CF6GM1 57391684 Ki = 1090 nM T60182 CM20FQ 57391685 Ki = 1450 nM T60182 CZ07MU 57391686 Ki = 12 nM T60182 CQ83PU 57392671 IC50 = 44 nM T60182 C5E9TH 57393252 IC50 = 19 nM T60182 CE8IH1 57393253 IC50 = 7.7 nM T60182 C8EJ5B 57393262 IC50 = 42 nM T60182 CW4FM5 57393425 Ki = 19 nM T60182 C7T0OK 57393426 Ki = 9 nM T60182 C03QCP 57394374 IC50 = 26 nM T60182 CYZX04 57396138 IC50 = 52 nM T60182 CB1V8N 57396139 IC50 = 34 nM T60182 CSQR94 57396140 IC50 = 17 nM T60182 CA29QU 57396141 IC50 = 17 nM T60182 CGI24C 57396925 Ki = 14700 nM T60182 C9M5VQ 57396926 Ki = 600 nM T60182 CUTF07 57396927 Ki = 1980 nM T60182 CIU91X 57396928 Ki = 91 nM T60182 COMA47 57397956 IC50 = 55 nM T60182 CS60YV 57397957 IC50 = 42 nM T60182 CUK67S 57399593 IC50 = 31 nM T60182 CS7VE8 57399594 IC50 = 9.2 nM T60182 CY4N6T 57400189 IC50 = 38 nM T60182 CBK59F 57400348 Ki = 1190 nM T60182 COPD34 57401358 IC50 = 51 nM T60182 C0FUB9 57401359 IC50 = 12 nM T60182 CAF67C 57401963 IC50 = 14 nM T60182 CDEQ30 57401986 IC50 = 1.7 nM T60182 CX68NH 57402151 Ki = 1110 nM T60182 C7HS2Q 57402152 Ki = 968 nM T60182 C7ZGC2 57402153 Ki = 556 nM T60182 C1KP5J 57403109 IC50 = 20 nM T60182 C4AJ1G 57403703 IC50 = 31 nM T60182 CK69YN 57403704 IC50 = 19 nM T60182 COK06F 57403898 Ki = 2160 nM T60182 C4WM0U 57518490 IC50 = 11.9 nM T60182 CJ9V0P 57882748 IC50 = 50 nM T60182 C81UIB 58352762 IC50 = 520 nM T60182 CLW17X 58352803 IC50 = 21 nM T60182 CTBN85 58352821 IC50 = 67 nM T60182 CX83MS 58352834 IC50 = 360 nM T60182 CQ6S2F 58352836 IC50 = 510 nM T60182 C7ODG8 58352840 IC50 = 1600 nM T60182 CFC36Q 58352858 IC50 = 490 nM T60182 CXF21H 58352863 IC50 = 85 nM T60182 C2I6KW 58352868 IC50 = 890 nM T60182 CYXQ05 58352925 IC50 = 340 nM T60182 CG4ZO9 58352935 IC50 = 170 nM T60182 C9M3WT 58352937 IC50 = 31 nM T60182 C2FN1G 58352938 IC50 = 5100 nM T60182 CW1UI5 58352940 IC50 = 720 nM T60182 CG3RK7 58352952 IC50 = 95 nM T60182 C12TUG 58352954 IC50 = 470 nM T60182 C7TG6Q 58352961 IC50 = 770 nM T60182 CH8MG0 58353013 IC50 = 96 nM T60182 C94ITK 58353025 IC50 = 340 nM T60182 C5PBI4 58353046 IC50 = 130 nM T60182 C3GQ6I 58353063 IC50 = 6 nM T60182 C9XR2K 58353067 IC50 = 23 nM T60182 CBH52R 58353104 IC50 = 220 nM T60182 CJ9F3R 58353126 IC50 = 10 nM T60182 C5UF0N 58353132 IC50 = 520 nM T60182 C5IXS0 58353156 IC50 = 480 nM T60182 COCJ18 58353206 IC50 = 82 nM T60182 CEFP60 58353232 IC50 = 940 nM T60182 CR1GW5 58353266 IC50 = 6800 nM T60182 CFBO93 58353274 IC50 = 3200 nM T60182 CX95LQ 58353323 IC50 = 13 nM T60182 C3KRI7 58353338 IC50 = 13 nM T60182 C1YPO0 58353350 IC50 = 620 nM T60182 C0SL8G 58353369 IC50 = 150 nM T60182 C9UW2R 58353408 IC50 = 1900 nM T60182 CR7UH2 58353464 IC50 = 1900 nM T60182 CU5D3M 58353489 IC50 = 800 nM T60182 CB9L4I 58353544 IC50 = 140 nM T60182 CD57RC 58353625 IC50 > 10000 nM T60182 CMLO57 58353662 IC50 = 44 nM T60182 CA7SI2 58353679 IC50 = 330 nM T60182 C1IND2 58353695 IC50 = 170 nM T60182 CLEZ12 58353778 IC50 = 1100 nM T60182 CG39KD 58353838 IC50 = 7 nM T60182 CO0ZG7 58353839 IC50 = 120 nM T60182 CU8GP5 58353901 IC50 = 730 nM T60182 C80TXA 58653097 IC50 = 303 nM T60182 CBM24G 59091612 IC50 = 6.9 nM T60182 CMZI93 59092268 IC50 = 221 nM T60182 CW17DA 60150962 Ki = 4100 nM T60182 C3EU9T 60151375 Ki = 890 nM T60182 C7XT6L 60151654 Ki = 700 nM T60182 CG4F9Z 60151793 Ki = 1100 nM T60182 C0UI2F 60151935 Ki = 1300 nM T60182 CKI5G1 60151936 Ki = 720 nM T60182 CH69GT 60151937 Ki = 1400 nM T60182 CO8W2J 60151938 Ki = 549 nM T60182 CPRV83 60152081 Ki = 1600 nM T60182 CT5X7B 60152219 Ki = 200 nM T60182 C1Z8WH 60152349 Ki = 100 nM T60182 C7E4ZQ 60152477 Ki = 170 nM T60182 C2FAN8 60152600 Ki = 160 nM T60182 CXC9I4 60152601 Ki = 12 nM T60182 C7FGW3 60152733 Ki = 220 nM T60182 CUD4H0 60152737 Ki = 1100 nM T60182 C68VYN 60152878 Ki = 1900 nM T60182 C1FKB3 60152880 Ki = 1700 nM T60182 CMJ51R 60170765 IC50 = 527.5 nM T60182 C9CLJ3 60170766 IC50 = 233.6 nM T60182 CYUG59 60170767 IC50 = 100.7 nM T60182 CK98DW 60170768 IC50 = 15.6 nM T60182 CTM07A 60170854 IC50 = 77.5 nM T60182 C6IV0K 60170855 IC50 = 16 nM T60182 CSN5C8 60170856 IC50 = 4.6 nM T60182 C4MKG9 60170857 IC50 = 13.3 nM T60182 CI59XA 60170968 IC50 = 15.3 nM T60182 CX7K6V 60170969 IC50 = 81.8 nM T60182 CPLU74 60170970 IC50 = 7.5 nM T60182 CX19CT 60170971 IC50 = 5.2 nM T60182 CA0EO3 60171059 IC50 = 1.9 nM T60182 C5JLE4 60171060 IC50 = 14.8 nM T60182 CQ6O3H 60171061 IC50 = 6.9 nM T60182 C2H1OF 60171062 IC50 = 9.3 nM T60182 CGEY07 68156267 Ki = 64 nM T60182 C20BGU 68156402 Ki = 5.6 nM T60182 CW42OI 68156701 Ki = 680 nM T60182 CIN8B5 68156716 Ki = 420 nM T60182 CI1EC3 68157252 Ki = 290 nM T60182 CLT25X 68178607 Ki = 4400 nM T60182 CDR1E8 68178611 Ki = 4100 nM T60182 C7YQK9 68178613 Ki = 230 nM T60182 C1K9MN 68186290 Ki = 1100 nM T60182 CX5FQ8 68243839 IC50 = 26 nM T60182 C3YW1K 68860750 IC50 = 292 nM T60182 CN2A8O 70695695 IC50 = 7.4 nM T60182 C3XY5M 70697675 IC50 = 21.2 nM T60182 CIV6E4 70900317 IC50 = 160 nM T60182 C76YUV 71060230 Ki = 33 nM T60182 CT9DV6 71202679 IC50 = 850 nM T60182 C85ZLB 71202712 IC50 = 370 nM T60182 CCY0M6 71202713 IC50 = 149 nM T60182 CM4R1O 71202743 IC50 = 230 nM T60182 C90NQH 71203427 IC50 = 190 nM T60182 CA69XP 71239397 Ki = 14 nM T60182 CND47O 71239512 Ki = 53 nM T60182 CF5WP9 71243005 IC50 = 24 nM T60182 C6DQ1U 71243036 IC50 = 100 nM T60182 C1K5TQ 71243097 IC50 = 180 nM T60182 CR42UV 71450867 IC50 = 61.8 nM T60182 CN9OP7 71452715 IC50 = 163 nM T60182 CFT42N 71454981 IC50 = 337.4 nM T60182 CBEL63 71456151 IC50 = 12.9 nM T60182 CN0G5Z 71456188 Ki > 500000 nM T60182 CSD43G 71614312 Ki = 670 nM T60182 CLIQ69 71614522 Ki = 170 nM T60182 CDX2U9 71614523 Ki = 6500 nM T60182 CF3X4N 73355438 IC50 = 671.43 nM T60182 C8SYW7 73355439 IC50 = 1230.27 nM T60182 C1WTZ8 90655064 IC50 = 1200 nM T60182 C9U1WM 90655065 IC50 = 65 nM T60182 CR26KU 90655066 IC50 = 1600 nM T60182 C1ON5Z 90655067 IC50 > 10000 nM T60182 CI6HW9 91755011 IC50 = 0.24 nM T60182 CN1HS8 122189569 IC50 = 26 nM T60182 C4SL9G 122189570 IC50 = 4 nM T60182 C37JMQ 122189571 IC50 = 1700 nM T60182 C5WFJ7 122189572 IC50 = 7 nM T60182 C58QDH 122189573 IC50 = 2 nM T60182 CKMW92 122189574 IC50 = 780 nM T60182 CC5L9Q 122189575 IC50 = 8 nM T60182 CUA94Z 122189576 IC50 = 4 nM T60182 CB53RK 122189577 IC50 = 1 nM T60182 CK5G1O 122189578 IC50 = 360 nM T60182 CO5IV3 122189579 IC50 = 7 nM T60182 CQ0WJ1 122189580 IC50 = 3 nM T60182 CN5G7Q 122189581 IC50 = 37 nM T60182 CG0T2V 122189693 IC50 = 5 nM T60182 CHW01S 122189694 IC50 = 10 nM T60182 C1TO8S 122189695 IC50 = 7 nM T60182 CXSR14 122189696 IC50 = 2 nM T60182 C08RBU 122189697 IC50 = 760 nM T60182 CEM9V2 122189698 IC50 = 50 nM T60182 C3NK1O 122189699 IC50 = 26 nM T60182 C9JNU4 122189700 IC50 = 72 nM T60182 CHLP75 122189701 IC50 = 8 nM T60182 CNY6K0 122189702 IC50 = 3 nM T60182 C3CPB4 122189703 IC50 = 4 nM T60182 C25XHS 122189704 IC50 = 6 nM T60182 CSB38V 122189705 IC50 = 15 nM T60182 C0DOI6 122189706 IC50 = 40 nM T60182 C8F4NT 122189707 IC50 = 35 nM T60182 CDAO27 122189708 IC50 = 1.9 nM T60182 CEQ09Z 122189709 IC50 = 2.6 nM T60182 CMAC12 122189710 IC50 = 1.5 nM T60182 CUIJ37 122189711 IC50 = 3 nM T60182 C9FBM1 122189712 IC50 = 18 nM T60182 C75EVN 122189713 IC50 = 1.5 nM T60182 CS1D9R 122189714 IC50 = 8 nM T60182 CWT0A5 122189715 IC50 = 1.6 nM T60182 C51BAG 122189716 IC50 = 3.4 nM T60182 C0WO4H 122189717 IC50 = 7 nM T60182 CT16NQ 122189718 IC50 = 18 nM T60182 CJO8I6 122189719 IC50 = 3.5 nM T60182 CE01SL 122189720 IC50 = 4 nM T60182 C5J4LM 122189721 IC50 = 4 nM T60182 CL0AR4 122189722 IC50 = 2.6 nM T60182 C3L5HZ 122189723 IC50 = 39 nM T60182 C7EAG8 122190361 Ki = 26 nM T60182 CH2LY9 122190362 Ki = 30 nM T60182 CL1J8A 122190363 IC50 = 4 nM T60182 COU48E 127045652 IC50 = 8900 nM T60182 C73SKL 127046098 IC50 = 1200 nM T60182 CZ6IR9 127046099 IC50 = 1500 nM T60182 C5U4SB 127046643 IC50 = 6300 nM T60182 C0I2QD 127046644 IC50 = 13000 nM T60182 C2D9UF 127046645 IC50 = 1900 nM T60182 C8TEO2 127046805 IC50 = 20800 nM T60182 C82VUJ 127046968 IC50 = 1200 nM T60182 CFZH26 127047120 IC50 = 6300 nM T60182 CSZV30 127047121 IC50 = 11100 nM T60182 CPT0N2 127047122 IC50 = 14500 nM T60182 C63SHZ 127047253 IC50 = 1400 nM T60182 C3UIJ1 127047254 IC50 = 10800 nM T60182 C6B5LM 127047255 IC50 = 5300 nM T60182 C6XR8O 127047256 IC50 = 2600 nM T60182 CE83XZ 127047385 IC50 = 2100 nM T60182 C6M4CR 127047904 IC50 = 1600 nM T60182 COW7R0 127047905 IC50 = 131100 nM T60182 CBLF95 127047906 IC50 = 26500 nM T60182 CEO7M5 127047907 IC50 = 4500 nM T60182 CH50JM 134304074 Ki = 29 nM T60182 CK70EH 134304075 Ki = 1850 nM T60182 C7PAK2 134304077 Ki = 144 nM T60182 CK7B0U 134304087 Ki = 23 nM T60182 CZ82QJ 134304088 Ki = 22 nM T60182 C6WD9T 134304090 Ki = 35 nM T60182 C63HEG 134304091 Ki = 22 nM T60182 CRFY98 134304096 Ki = 35 nM T60182 CX62UZ 134304119 Ki = 32 nM T60182 CUDY24 134304129 Ki = 14 nM T60182 CUP03B 134304131 Ki = 36 nM T60182 CIM48Y 134304136 Ki = 125 nM T60182 C6FSP7 134304141 Ki = 100 nM T60182 CPC91L 134304142 Ki = 114 nM T60182 C3XG8V 134304145 Ki = 85 nM T60182 C7EU6S 134304147 Ki = 86 nM T60182 CA8C5Z 134304151 Ki = 150 nM T60182 CA8RS4 134304160 Ki = 115 nM T60182 C1P6FK 134304171 Ki = 30 nM T60182 COZ3S0 134304173 Ki = 57 nM T60182 CO5I4B 134304177 Ki = 25 nM T60182 CR6NL4 134304181 Ki = 86 nM T60182 CO3QR9 134304190 Ki = 42 nM T60182 C9A3PS 134304191 Ki = 650 nM T60182 CS4CF9 134304192 Ki = 32 nM T60182 CO9SD3 134304194 Ki = 175 nM T60182 CE7HI9 134304208 Ki = 1269 nM T60182 C6U3TO 134304209 Ki = 100 nM T60182 CH8T2K 134304219 Ki = 44 nM T60182 C4ULW3 134304232 Ki = 2800 nM T60182 CK84WL 134304234 Ki = 22 nM T60182 CX27VI 134304713 Ki = 115 nM T60182 C5TU3S 134304793 Ki = 700 nM T60182 C64TDW 134304822 Ki = 85 nM T60182 C9VHO5 134304824 Ki = 110 nM T60182 CR2F3W 134309610 Ki = 125 nM T60182 CZ10SK 135407749 IC50 > 100000 nM T60182 CU64IB 135427275 IC50 > 100000 nM T60182 CUM29I 135437141 IC50 = 60000 nM T60182 C4QYH6 135442286 IC50 = 3400 nM T60182 C7ZW8M 135443742 IC50 > 100000 nM T60182 C5SO9D 135447739 IC50 > 100000 nM T60182 C5MCS9 135451009 IC50 > 100000 nM T60182 C80OZY 135470359 IC50 > 100000 nM T60182 C90GUW 135470389 IC50 = 720 nM T60182 C0AM7Y 135471545 IC50 > 100000 nM T60182 CU7C2P 135501650 IC50 = 28000 nM T60182 CZ0CO5 135503676 IC50 = 200 nM T60182 CG7LX6 135503833 Ki > 500000 nM T60182 CN0OI8 135503932 Ki > 500000 nM T60182 CNF57J 135504174 IC50 = 23000 nM T60182 C1USI4 135533241 IC50 = 390 nM T60182 CI16PU 135538097 IC50 > 100000 nM T60182 CK1E7J 135538098 IC50 = 2000 nM T60182 C7HEG5 135542439 IC50 = 1200 nM T60182 C6C0YG 135542465 IC50 = 34000 nM T60182 CI82RJ 135542514 IC50 > 100000 nM T60182 CX50HZ 135542516 IC50 > 100000 nM T60182 CYD2O9 135544439 IC50 = 830 nM T60182 CA2FR5 135545151 IC50 > 100000 nM T60182 CGP2W3 135819133 IC50 = 12 nM T60182 C0U6JN 135819135 IC50 = 500 nM T60182 C2H1YV 135819137 IC50 = 120 nM T60182 CCOB80 135819143 IC50 = 28 nM T60182 C4ENV0 135819146 IC50 = 10 nM T60182 C8C2OQ 135819149 IC50 = 40 nM T60182 CRG7M0 135819157 IC50 = 16 nM T60182 CAQ82J 136055807 IC50 = 5200 nM T60182 CX5MS9 137633159 EC50 = 0.0062 nM T60182 C3YHG5 137634214 EC50 = 0.0156 nM T60182 CY40VR 137634741 EC50 = 2.32 nM T60182 CB4I7O 137638423 EC50 = 1.24 nM T60182 CEX6K4 137642925 EC50 = 0.0007 nM T60182 CQ7E1C 137643772 EC50 = 0.0089 nM T60182 CK2JM7 137649897 EC50 = 0.0019 nM T60182 CI72XO 137650720 EC50 = 1.12 nM T60182 CS8WM2 137654780 EC50 = 0.0063 nM T60182 C5ZD1M 137659233 EC50 = 0.0264 nM T60182 CZK81P 137661599 EC50 = 0.008 nM T60182 CJ5FS6 137662302 EC50 = 0.12 nM T60182 C1C4YM 141465319 IC50 = 550 nM T60182 C1GTU0 141465320 IC50 = 800 nM T60182 C8WFD2 141465324 IC50 = 100 nM T60182 C7LUP2 141465337 IC50 = 4920 nM T60182 C5EGJ9 141465346 IC50 = 830 nM T60182 CQ29TZ 145949291 EC50 = 1.57 nM T60182 C4LE9A 145949559 EC50 = 3.88 nM T60182 CB8O0I 145950198 EC50 = 2.81 nM T60182 C8K1TP 145950470 EC50 = 18.64 nM T60182 CIFH84 145951037 EC50 = 0.86 nM T60182 CG52YC 145952042 EC50 = 3.36 nM T60182 CV0C2K 145952411 EC50 = 0.75 nM T60182 C7MC0S 145953388 EC50 = 1.27 nM T60182 CGLY87 145953555 EC50 = 0.9 nM T60182 C9A1LQ 145953718 EC50 = 2.4 nM T60182 C7CK8M 145953834 EC50 = 1.43 nM T60182 C3A6GO 145956482 EC50 = 6.99 nM T60182 CHP34N 145956533 EC50 = 122.57 nM T60182 C6OFU3 145956601 EC50 = 4.49 nM T60182 CW5PY0 145956908 EC50 = 1.41 nM T60182 C0M6PJ 145957642 EC50 = 4.78 nM T60182 CLKX02 145958107 EC50 = 5.3 nM T60182 C96YSZ 145958355 EC50 = 1.41 nM T60182 CSQ0B2 145958772 EC50 = 0.46 nM T60182 CGNW71 145959528 EC50 = 2.84 nM T60182 CW1X9P 145959606 EC50 = 14.6 nM T60182 C7HZY1 145959966 EC50 = 1.29 nM T60182 C7N3KL 145960401 EC50 = 0.0025 nM T60182 C92BLJ 145960433 EC50 = 0.0019 nM T60182 C0X5MI 145960850 EC50 = 0.029 nM T60182 CT1JB9 145961416 EC50 = 4.37 nM T60182 C1ZNU5 145961751 EC50 = 0.0016 nM T60182 CW90YV 145962263 EC50 = 42.9 nM T60182 CN9CR1 145962270 EC50 = 0.0044 nM T60182 CA29XQ 145962515 EC50 = 0.0154 nM T60182 CVQ62L 145962554 EC50 = 0.0276 nM T60182 C97HKT 145962593 EC50 = 0.0007 nM T60182 CGO8V1 145962872 EC50 = 0.0067 nM T60182 C0ADY2 145962907 EC50 = 3.09 nM T60182 CXFC81 145967583 IC50 = 740 nM T60182 CLO0S4 145967618 EC50 = 5.225 nM T60182 C8D7VX 145967685 IC50 = 220 nM T60182 C8IZ5K 145967741 IC50 = 630 nM T60182 C47SXA 145967899 IC50 = 2310 nM T60182 C1VY2O 145967924 IC50 = 310 nM T60182 CQDI82 145967926 EC50 > 1000 nM T60182 CUAD30 145968045 IC50 = 70 nM T60182 C83TNS 145968140 IC50 = 3230 nM T60182 CUQD98 145968206 IC50 = 1920 nM T60182 C3JW1P 145968295 EC50 = 0.041 nM T60182 C0T1ZE 145968501 EC50 = 0.005 nM T60182 C0ZTW8 145968513 EC50 = 0.005 nM T60182 CMB10N 145969232 EC50 = 0.006 nM T60182 C4L1VQ 145969278 IC50 = 570 nM T60182 C5J8HP 145969289 EC50 = 0.03 nM T60182 C2D4EA 145969298 IC50 = 110 nM T60182 CLJ78O 145969316 IC50 = 230 nM T60182 CZ79BS 145969571 IC50 = 300 nM T60182 C7UZT9 145969722 EC50 = 0.028 nM T60182 CS36QG 145969945 EC50 = 0.031 nM T60182 CTA7Z5 145969968 IC50 = 180 nM T60182 C3AI9B 145970440 EC50 = 0.15 nM T60182 CX0C6A 145970613 EC50 = 0.009 nM T60182 CCZ9K7 145970869 EC50 = 0.007 nM T60182 C3XI1H 145970930 IC50 = 80 nM T60182 CO3DS8 145970933 IC50 = 2790 nM T60182 CDNQ48 145971078 IC50 = 370 nM T60182 CDB15L 145971098 EC50 = 0.016 nM T60182 CB0IC1 145971123 IC50 = 500 nM T60182 CN4Z2C 145971132 EC50 = 0.004 nM T60182 CV4F0E 145974582 EC50 = 2.99 nM T60182 CY3OT1 145981450 IC50 = 6900 nM T60182 C8RD2J 145982299 IC50 = 8200 nM T60182 C7GP9V 145986381 IC50 = 9300 nM T60182 C2J1OP 145986774 IC50 = 17700 nM T60182 CC3Y2Z 145987495 EC50 = 0.003 nM T60182 CD5A9X 145989050 IC50 = 60 nM T60182 CPG4M5 145989480 IC50 = 3900 nM T60182 C7W4UH 145989947 IC50 = 6000 nM T60182 CU2HL7 145990090 IC50 = 4100 nM T60182 CAE9L4 145993424 IC50 = 8500 nM T60182 CE2MR1 155512720 EC50 = 0.0843 nM T60182 CT04BK 155515237 Ki = 1250 nM T60182 CDYC28 155515554 Ki = 19 nM T60182 CJD32Q 155517094 EC50 = 0.0714 nM T60182 CWY0N7 155517246 Ki = 255 nM T60182 CT6YU8 155523482 EC50 = 0.017 nM T60182 CV8L5S 155526074 Ki = 1345 nM T60182 CM2Z6O 155526545 EC50 = 0.0359 nM T60182 CA18CO 155528087 Ki = 3000 nM T60182 CPIU28 155530534 Ki = 199 nM T60182 CEM4C1 155532070 EC50 = 2.325 nM T60182 CN25WB 155532202 EC50 = 0.0309 nM T60182 CYPT96 155533592 EC50 = 0.0268 nM T60182 C2EJR8 155536703 Ki = 460 nM T60182 C46ZGV 155538812 Ki = 1100 nM T60182 C10BXG 155539799 Ki = 1350 nM T60182 C6WAG2 155541176 Ki = 285 nM T60182 CKI6O4 155543961 EC50 > 0.001 nM T60182 CO59AZ 155549801 Ki = 96 nM T60182 C0JZE8 155555973 Ki = 800 nM T60182 C9JK7Y 155558364 Ki = 1650 nM T60182 CA6MK0 155560326 Ki > 2600 nM T60182 CT1S6B 155562429 EC50 = 0.0339 nM T60182 C56IJU 155564592 EC50 = 0.0399 nM T60182 CSFY13 155566739 EC50 = 0.0379 nM T60182 D04IUW 44584360 IC50 = 440 nM T60182 D08XLL 619101 IC50 = 129 nM T60182 D0I6HV 4206177 Ki = 20000 nM T60182 D0M3AR 5311276 IC50 = 7 nM T60182 D0VC0I 5169 IC50 = 80.17 nM T59554 CYL3G4 390818 IC50 = 41 nM T59554 CSXL49 390820 IC50 = 72 nM T59554 CQZ2A9 16423013 IC50 = 70 nM T59554 CN30PZ 45606653 IC50 = 1584.89 nM T59554 C3RJ0P 45606655 IC50 = 1258.93 nM T59554 CFOD38 47056816 IC50 = 794.33 nM T59554 CX8JP5 67402849 IC50 > 10000 nM T59554 CT23SN 86287487 IC50 = 120 nM T59554 C05VLX 86287489 IC50 = 88 nM T59554 C8G1XP 86287490 IC50 = 80 nM T59554 CTH2B9 86287491 IC50 = 50 nM T59554 CX3P5J 86287492 IC50 = 67 nM T59554 CG7T0R 86582124 IC50 = 100 nM T59554 CBF8L1 118569872 IC50 = 9600 nM T59554 CMO32D 121465021 IC50 > 10000 nM T59554 CE7H5V 121465028 IC50 = 60 nM T59554 CHO8N2 129901999 IC50 < 8000 nM T59554 CK8L1S 129902000 IC50 < 8000 nM T59554 CM4Q9A 129902199 IC50 < 8000 nM T59554 CVW5X0 155510774 IC50 = 19952.62 nM T59554 C8WTR6 155511153 IC50 = 3981.07 nM T59554 CG4UR8 155513177 IC50 = 501.19 nM T59554 C7L4TB 155513385 IC50 = 79.43 nM T59554 CZ23GQ 155514135 IC50 = 31.62 nM T59554 C4JX1E 155514986 IC50 = 63.1 nM T59554 CEP9R6 155515121 IC50 = 1258.93 nM T59554 C2URD1 155515364 IC50 = 100000 nM T59554 CP1Z2N 155515497 IC50 = 63.1 nM T59554 CZ7D6C 155516581 IC50 = 100 nM T59554 C1KIG4 155517111 IC50 = 501.19 nM T59554 CJ85TL 155517302 IC50 = 794.33 nM T59554 CA13KU 155518587 IC50 = 1995.26 nM T59554 COR3P1 155520360 IC50 = 7943.28 nM T59554 CU2MR9 155520898 IC50 = 794.33 nM T59554 CAQX37 155521638 IC50 = 1800 nM T59554 CWCN51 155522922 IC50 = 30 nM T59554 CAL9M0 155523067 IC50 = 79.43 nM T59554 CW6VR0 155523250 IC50 = 10000 nM T59554 C5RHS4 155523529 IC50 = 199.53 nM T59554 CEGX23 155523680 IC50 = 199.53 nM T59554 C81SMD 155525007 IC50 = 3162.28 nM T59554 C9R5LH 155525273 IC50 = 158.49 nM T59554 CM9F1U 155525433 IC50 = 630.96 nM T59554 CQ39FV 155525552 IC50 = 2511.89 nM T59554 C7D4PR 155526164 IC50 = 10000 nM T59554 C6L8SR 155526637 IC50 = 5011.87 nM T59554 CLP34R 155526851 IC50 = 398.11 nM T59554 CNH0S3 155526984 IC50 < 8000 nM T59554 CL8Z3K 155527451 IC50 = 100 nM T59554 C84PYB 155527664 IC50 = 31622.78 nM T59554 C0IK2N 155527755 IC50 = 79.43 nM T59554 CAS9F3 155529191 IC50 = 1000 nM T59554 C9HG5P 155529534 IC50 = 630.96 nM T59554 C7R9KJ 155530796 IC50 = 158.49 nM T59554 CIU3J0 155532031 IC50 = 2511.89 nM T59554 C62FTB 155532792 IC50 = 158.49 nM T59554 C50SOB 155532814 IC50 = 251.19 nM T59554 C6R8JM 155533521 IC50 = 79.43 nM T59554 C7TZP5 155534028 IC50 = 794.33 nM T59554 CW5VE8 155534801 IC50 = 100 nM T59554 CI02AF 155535182 IC50 = 316.23 nM T59554 CP8WA7 155535854 IC50 = 1258.93 nM T59554 CHT4R0 155538088 IC50 = 501.19 nM T59554 CTU90R 155539548 IC50 = 31622.78 nM T59554 CL3V4X 155540013 IC50 = 125.89 nM T59554 C47FDX 155542118 IC50 = 630.96 nM T59554 CW1KR5 155544065 IC50 = 5011.87 nM T59554 C46WQE 155545645 IC50 = 79432.82 nM T59554 CT4X7K 155545722 IC50 = 3162.28 nM T59554 C58XCM 155550370 IC50 = 398.11 nM T59554 CL5WO0 155551218 IC50 = 6309.57 nM T59554 C2BQR9 155551582 IC50 = 630.96 nM T59554 C7NR3U 155554730 IC50 = 79.43 nM T59554 CS97XD 155555252 IC50 = 1000 nM T59554 CIQW10 155555500 IC50 = 25118.86 nM T59554 CQA79R 155555533 IC50 = 1995.26 nM T59554 C8EIB2 155556353 IC50 = 199.53 nM T59554 CYJQ95 155556388 IC50 = 630.96 nM T59554 C7AZ5J 155556578 IC50 = 63.1 nM T59554 CNI2B8 155556601 IC50 = 6309.57 nM T59554 CSCZ69 155556758 IC50 = 63.1 nM T59554 CZ78PF 155559436 IC50 = 25118.86 nM T59554 CJ32XC 155560820 IC50 = 158.49 nM T59554 CTL04N 155562816 IC50 = 199.53 nM T59554 CD5FO3 155567866 IC50 = 199.53 nM T59554 CQ59SD 155568558 IC50 = 5011.87 nM T59554 CUQ9R8 155569026 IC50 = 63.1 nM T59554 C2DZ5S 155569117 IC50 = 12589.25 nM T59554 C12YCW 155569543 IC50 = 100 nM T59554 CQHA48 155569656 IC50 = 7943.28 nM T99009 D00HGB 4488 IC50 = 17000 nM T99009 D08ROP 3899 IC50 = 10000 nM T99009 D09SOA 28718 IC50 = 13000 nM T99009 D00LSI 9820008 IC50 = 134 nM T99009 D0G7UX 5284373 IC50 > 50000 nM T99009 D0N3XT 57030 IC50 = 6 nM T99009 CYIU47 1543 IC50 = 7 nM T99009 CI9TK0 3884 IC50 = 100 nM T99009 CR6HO1 8593 IC50 = 144000 nM T99009 CU4O3D 38081 IC50 = 8000 nM T99009 C5LA7B 76864 IC50 = 709 nM T99009 CE2KN9 130331 Ki = 25 nM T99009 CYRV23 131419 IC50 = 12 nM T99009 CS74HZ 145726 IC50 = 12380 nM T99009 C4U5MD 202918 IC50 = 10000 nM T99009 C21UMY 271388 IC50 = 541 nM T99009 CT6MA7 322307 IC50 > 10000 nM T99009 CP4ZX0 459316 IC50 = 420 nM T99009 CVY91W 517728 IC50 > 100000 nM T99009 CEVD28 517858 IC50 > 100000 nM T99009 C9JAF2 523003 IC50 > 200000 nM T99009 CO0MN5 609454 IC50 > 20000 nM T99009 CZH54C 615334 IC50 > 20000 nM T99009 C14CXW 619026 IC50 = 3960 nM T99009 CJ1W4Q 623973 IC50 = 3410 nM T99009 COPS41 653193 IC50 > 100000 nM T99009 CDX0O4 660996 IC50 > 200000 nM T99009 CXS49M 669445 IC50 = 6830 nM T99009 CZO9S8 673239 IC50 = 13010 nM T99009 C4UOR0 673730 IC50 = 5176.8 nM T99009 CCLM40 684865 IC50 = 930 nM T99009 CG2Q8Y 736801 IC50 = 18280 nM T99009 C5UJV1 739902 IC50 = 1830 nM T99009 C8S6ZO 741601 IC50 > 100000 nM T99009 C23WHO 741604 IC50 > 100000 nM T99009 C76COZ 743061 IC50 > 200000 nM T99009 CFD56M 753240 IC50 = 1566.1 nM T99009 CE6G1W 777184 IC50 > 100000 nM T99009 CS4BA6 777191 IC50 > 100000 nM T99009 CFD0U2 780529 IC50 = 17750 nM T99009 C4GAY3 813108 IC50 = 15620 nM T99009 C2PSU0 831397 IC50 = 780 nM T99009 CC4S8F 844231 IC50 = 550 nM T99009 CC0MD2 865225 Ki > 500 nM T99009 CIQ10J 904019 IC50 = 3249.8 nM T99009 CH52WR 947453 IC50 = 9074 nM T99009 CBT92O 993994 IC50 = 136.2 nM T99009 CSBU38 1027581 IC50 = 1270 nM T99009 C9JCR6 1037067 IC50 = 340 nM T99009 CQYE56 1133093 IC50 = 5900 nM T99009 C3O5MX 1223586 IC50 = 57.1 nM T99009 C87PLH 1223597 IC50 = 666.2 nM T99009 C8HS9K 1374134 IC50 = 1130 nM T99009 COV67N 1432578 IC50 = 400 nM T99009 CG1F9T 1460771 IC50 > 100000 nM T99009 CM4L5I 1481799 IC50 = 17400 nM T99009 C1KT8C 1746237 IC50 = 260 nM T99009 CR3IN2 1746284 IC50 = 1310 nM T99009 CGDC52 1763612 IC50 = 436.7 nM T99009 C5S6NK 1830299 IC50 = 250 nM T99009 CYA5F2 1965647 IC50 = 89000 nM T99009 C8NMY3 2063288 IC50 = 51 nM T99009 C93GMJ 2578400 IC50 > 20000 nM T99009 C9HOI8 2709135 IC50 = 12400 nM T99009 C31KAP 2743369 IC50 = 39000 nM T99009 C7GE9J 2759386 IC50 = 1040 nM T99009 CH25IU 2858282 IC50 > 10000 nM T99009 CS0KO4 2995335 IC50 = 16080 nM T99009 CN0MT1 3100461 IC50 = 29 nM T99009 CX2L9S 3227262 IC50 > 100000 nM T99009 CS7MF9 3851642 Ki = 17900 nM T99009 C54XIU 3899945 IC50 = 1600 nM T99009 C01OYK 4221076 Ki = 35900 nM T99009 CR9A1Q 4605417 IC50 > 500000 nM T99009 C8JYO2 4749758 IC50 = 3848 nM T99009 CMSE21 5057449 IC50 = 9.7 nM T99009 C1TC3N 5167181 Ki = 28 nM T99009 CJ1BM6 5184531 IC50 > 200000 nM T99009 CU73XG 5287459 Ki = 2800 nM T99009 CK86XL 5308416 IC50 > 100000 nM T99009 CYP02U 5376552 IC50 = 10000 nM T99009 CM4A3N 7346373 IC50 = 81 nM T99009 CNY5I0 7416167 IC50 > 100000 nM T99009 CE5XO9 7688340 IC50 = 1300 nM T99009 C67CZW 7955004 IC50 = 1358 nM T99009 C9KT2N 8850862 IC50 > 100000 nM T99009 C0LYE6 9045495 IC50 > 20000 nM T99009 C0KG4F 9173919 IC50 > 10000 nM T99009 CCGE73 9547914 IC50 = 280 nM T99009 CQ70AU 9824035 Ki = 4 nM T99009 CHZ34C 9861992 IC50 = 303 nM T99009 C0XCI6 9948506 IC50 = 410 nM T99009 CNP6S9 10000399 Ki = 13 nM T99009 CG7EM6 10029745 Ki = 26 nM T99009 CRA6E7 10048413 Ki = 4 nM T99009 CA7TO9 10064328 IC50 = 700 nM T99009 C1EF4U 10342449 IC50 = 33 nM T99009 CB4D0C 10356750 IC50 > 100000 nM T99009 CJ1KH3 10364016 Ki = 8.4 nM T99009 C3S6CZ 10404208 IC50 = 800 nM T99009 CIO0Z9 10454174 IC50 = 8 nM T99009 CZ4KA1 10457096 IC50 = 7 nM T99009 C68KRG 10488180 IC50 > 50000 nM T99009 C5ZE1V 10491179 IC50 = 3600 nM T99009 CI31FC 10492984 IC50 > 50000 nM T99009 C4N5YT 10494611 IC50 = 6060 nM T99009 CCFG07 10496492 IC50 > 50000 nM T99009 C6REV7 10512886 IC50 = 19400 nM T99009 COVK03 10515945 IC50 > 50000 nM T99009 CC1K4I 10516844 IC50 > 50000 nM T99009 CM15VH 10516983 IC50 = 500 nM T99009 CU5PT2 10519719 IC50 > 50000 nM T99009 C54GLO 10540764 IC50 = 6200 nM T99009 C54IJE 10541884 IC50 = 6500 nM T99009 C0PLE3 10544308 IC50 > 50000 nM T99009 C32DIH 10565707 IC50 = 4000 nM T99009 CED3A9 10565785 IC50 > 50000 nM T99009 CY1RS4 10587807 IC50 > 50000 nM T99009 CLXD24 10587934 IC50 > 50000 nM T99009 C42WEO 10635802 IC50 = 2700 nM T99009 CHDR60 10643787 Ki = 6000 nM T99009 C81RJI 10657722 IC50 = 16500 nM T99009 CZ4DH9 10680043 IC50 = 12100 nM T99009 C6ZNV5 10680597 IC50 = 3200 nM T99009 C4X0UR 10682218 IC50 = 22400 nM T99009 CQ96TA 10687946 Ki = 3700 nM T99009 CH1UQ6 10690749 Ki = 4000 nM T99009 C15GIF 10691466 Ki > 100000000 nM T99009 CI5AT8 10703799 IC50 > 50000 nM T99009 C21DPI 10710291 IC50 > 50000 nM T99009 C1H3PI 10711746 IC50 > 50000 nM T99009 CZQH50 10738106 Ki > 100000000 nM T99009 CIG1Q0 10752727 IC50 = 9000 nM T99009 CJ1ED3 10755169 IC50 > 50000 nM T99009 C27DHQ 10759123 IC50 > 50000 nM T99009 CU26LB 10759927 IC50 > 50000 nM T99009 CU29BN 10800984 IC50 = 22500 nM T99009 CX5EL6 10805428 IC50 > 50000 nM T99009 C6O0EX 10808375 IC50 = 239 nM T99009 CIW5B8 10825617 IC50 = 2600 nM T99009 CUZ3X1 10828593 IC50 > 50000 nM T99009 C3HM9N 10829333 IC50 > 50000 nM T99009 CDV5Q8 10830186 IC50 > 50000 nM T99009 CRZH97 10830342 Ki = 4000 nM T99009 CY53LI 10849345 IC50 > 50000 nM T99009 CBRS89 10852951 Ki = 20000 nM T99009 C3PU1H 10853437 IC50 = 784 nM T99009 C4VCG7 10895558 Ki = 32 nM T99009 CRJ4Q5 10929378 Ki = 331 nM T99009 C2Q8UR 10938858 Ki = 12 nM T99009 CV1KX4 11016730 Ki = 8 nM T99009 CL4CV9 11038663 Ki = 1500 nM T99009 C87CWY 11102808 Ki = 6 nM T99009 CVGQ92 11135071 Ki = 2400 nM T99009 CMW42X 11416123 Ki = 203 nM T99009 C1D5CH 11524688 IC50 = 1 nM T99009 C5IEU6 11530041 IC50 > 200000 nM T99009 C4C1QF 11703683 IC50 > 200000 nM T99009 CKS30M 11762691 Ki = 138 nM T99009 C6NY3W 11825758 Ki = 91 nM T99009 CUB8Y3 12454047 Ki = 15100 nM T99009 CE6Z4B 13960629 Ki = 60 nM T99009 COMT87 13960632 Ki = 29 nM T99009 CK5RC6 13960639 Ki = 30 nM T99009 C51BST 13960640 Ki = 20 nM T99009 C2GNU0 13960650 Ki = 10 nM T99009 C0UX8F 13960654 Ki = 13 nM T99009 CYJ08U 13960663 Ki = 220 nM T99009 C4XWV8 13960668 Ki = 10 nM T99009 C0QF9I 13960681 Ki = 270 nM T99009 C7T2LK 14222046 IC50 = 2800 nM T99009 CJQS85 14498146 IC50 = 5 nM T99009 CP17YT 14498150 IC50 = 10 nM T99009 CZ9B2W 14498162 IC50 = 312 nM T99009 CZ13DK 14498163 IC50 = 211 nM T99009 CU29XS 14498165 IC50 = 217 nM T99009 CXB50A 14498174 IC50 = 6 nM T99009 CW3P1R 14498175 IC50 = 7 nM T99009 CR7KX9 14498179 IC50 = 18 nM T99009 C1ORM4 14773532 Ki = 17 nM T99009 CL3M4G 15858807 IC50 > 50000 nM T99009 CQN40R 15942657 IC50 = 44 nM T99009 CP2WJ3 15942658 IC50 = 2 nM T99009 CXV7A5 16099894 IC50 = 306000 nM T99009 COH7N2 16099900 IC50 = 151000 nM T99009 C8D0KF 16099905 IC50 = 72000 nM T99009 CM8CL1 16099913 IC50 = 56000 nM T99009 C3UK7A 16099914 IC50 = 136000 nM T99009 C3V2KY 16099916 IC50 = 212000 nM T99009 CR5EY8 16099917 IC50 = 17000 nM T99009 CBE84I 16099918 IC50 = 51000 nM T99009 C31XCS 16099919 IC50 = 283000 nM T99009 C2FXW0 16099923 IC50 = 26000 nM T99009 CFY05L 16099926 IC50 = 230000 nM T99009 CO5SY7 16099929 IC50 = 4000 nM T99009 COSK93 16099935 IC50 = 135000 nM T99009 C51NZE 16099968 IC50 = 301000 nM T99009 C2NH3G 16099971 IC50 = 41000 nM T99009 C0IBF1 16099978 IC50 = 32000 nM T99009 C8HGF0 16100002 IC50 = 134000 nM T99009 CUM26S 16100003 IC50 = 141000 nM T99009 C4ZVE0 16100004 IC50 = 130000 nM T99009 CUMK61 16100005 IC50 = 270 nM T99009 CDG5U9 16100006 IC50 = 132000 nM T99009 CE39KU 16100011 IC50 = 43000 nM T99009 C7VE4W 16100015 IC50 = 4900 nM T99009 CJM54Z 16102641 Ki = 3630 nM T99009 CZX30A 16102642 Ki = 60400 nM T99009 CKT91D 16102643 IC50 > 500000 nM T99009 CMEU86 16102644 Ki = 27 nM T99009 COQW13 16102645 Ki = 12800 nM T99009 CL3A8Z 16102646 IC50 > 500000 nM T99009 CXO5U1 16210733 IC50 = 1440 nM T99009 CXUO14 16457485 IC50 = 46000 nM T99009 C83SPM 16457486 IC50 = 12000 nM T99009 C8MSK3 16777509 IC50 > 200000 nM T99009 CD20AH 21084669 IC50 = 42 nM T99009 CA9Z7Y 21084690 IC50 = 225 nM T99009 CI1T5W 21084721 IC50 = 170 nM T99009 C37ANI 21084723 IC50 = 45 nM T99009 CDS2T7 21084730 IC50 = 110 nM T99009 C1XP7M 21084734 IC50 = 90 nM T99009 CL46XF 21084739 IC50 = 310 nM T99009 C06TFS 21084741 IC50 = 11 nM T99009 C6XJ2K 21084746 IC50 = 8400 nM T99009 C58MIH 21084752 IC50 = 17 nM T99009 CI41ZH 21084760 IC50 = 1700 nM T99009 CHE52U 21084763 IC50 = 5700 nM T99009 C0B6YR 21084801 IC50 = 127 nM T99009 CK7N2M 21084803 IC50 = 2000 nM T99009 C1AW4H 21084857 IC50 = 105 nM T99009 CND19K 21084860 IC50 = 173 nM T99009 C38QSO 21084861 IC50 = 667 nM T99009 C6QYE9 22042531 IC50 = 680 nM T99009 C8RBW0 22042533 IC50 = 1460 nM T99009 CP09OF 22431257 IC50 > 100000 nM T99009 CK02UJ 22433941 IC50 > 100000 nM T99009 C0I8AV 22577320 IC50 > 100000 nM T99009 C09MTF 22579221 IC50 > 100000 nM T99009 C5AR8O 23647298 Ki > 100000000 nM T99009 CS0RU6 23647299 IC50 = 3 nM T99009 CZAT30 23647300 IC50 = 9 nM T99009 C29UME 23647301 IC50 = 12 nM T99009 C8Y6DJ 23647302 IC50 = 1000 nM T99009 CWFG85 23647303 IC50 = 10 nM T99009 C6GOR3 23647305 IC50 > 1000 nM T99009 CUJ9D8 23647306 IC50 > 1000 nM T99009 CQOP01 23647307 IC50 > 1000 nM T99009 C8GJ7K 23647308 IC50 = 16 nM T99009 C9AVR7 23647309 IC50 = 340 nM T99009 C3WMP9 23663733 Ki = 24 nM T99009 CG5YM6 23663964 Ki = 12 nM T99009 C7KBU5 23668107 Ki = 15 nM T99009 CQYE41 23668976 Ki = 8.3 nM T99009 CK7MW5 23671800 Ki = 40 nM T99009 CT3AJ5 23671801 Ki = 17 nM T99009 CN3FK4 23673359 Ki = 8 nM T99009 CP01FB 23673369 Ki = 38 nM T99009 CE9OD6 23673384 Ki = 24 nM T99009 CRK25G 23673385 Ki = 210 nM T99009 CR59ZP 23673428 Ki = 230 nM T99009 CT7XA2 23686481 Ki = 170 nM T99009 CB94XJ 23693316 Ki = 31 nM T99009 C1HEK3 23699178 Ki = 4.5 nM T99009 C5T0GQ 23699179 Ki > 130 nM T99009 C96KCH 23699180 Ki = 27 nM T99009 CR2KJ1 23699181 Ki = 26 nM T99009 CL3ZU5 23699195 Ki = 25 nM T99009 C2E0MI 23699196 Ki = 52 nM T99009 CWE6Z3 24829334 IC50 = 2.999 nM T99009 CJ3Z9A 24882111 IC50 > 200000 nM T99009 CZVG60 24882112 IC50 > 200000 nM T99009 CD26YW 24882113 IC50 > 200000 nM T99009 C4WDG1 24882114 IC50 > 200000 nM T99009 C5T0WI 24882115 IC50 > 200000 nM T99009 CO39XG 24882194 IC50 > 200000 nM T99009 C8RBY3 24882195 IC50 > 200000 nM T99009 CMW12Z 24882196 IC50 > 200000 nM T99009 C5YZR8 24882197 IC50 > 200000 nM T99009 C5QHJ4 24882198 IC50 > 200000 nM T99009 CYV89J 24986460 IC50 = 87.9 nM T99009 CUN1P0 24986824 IC50 = 15 nM T99009 C38QGT 24986825 IC50 = 19.01 nM T99009 C8WCI6 24986827 IC50 = 89.95 nM T99009 C5JQG2 24987180 IC50 = 149.97 nM T99009 C35LNQ 24987183 IC50 = 19.01 nM T99009 CJ03WL 24987187 IC50 = 14 nM T99009 CS62EF 24987532 IC50 = 199.99 nM T99009 CS4BW8 24987910 IC50 = 11.99 nM T99009 CP1R6W 24987911 IC50 = 99.08 nM T99009 CDR80K 24987915 IC50 = 109.9 nM T99009 CXB25G 24987916 IC50 = 11.99 nM T99009 CGZU50 24988290 IC50 = 32.96 nM T99009 CTG18W 24988292 IC50 = 5.998 nM T99009 CM2L0X 24988658 IC50 = 5 nM T99009 CG75AI 24988659 IC50 = 17.02 nM T99009 CD35ZG 24988663 IC50 = 52.97 nM T99009 CDEO28 24988664 IC50 = 23.01 nM T99009 C92RNP 24989025 IC50 = 3.999 nM T99009 CE3L9I 24989026 IC50 = 7.998 nM T99009 C06BXV 24989027 IC50 = 10.99 nM T99009 CN5ZM2 24989028 IC50 = 3.999 nM T99009 CY7L9T 24989029 IC50 = 5.998 nM T99009 CIY92Z 24989389 IC50 = 5 nM T99009 CHAV93 24991946 IC50 = 199.99 nM T99009 CDH5W8 25263414 IC50 > 100000 nM T99009 CB15SF 25263431 IC50 > 100000 nM T99009 CL3SD8 25263432 IC50 > 100000 nM T99009 C5Z3US 25263434 IC50 > 100000 nM T99009 COLC28 25495325 IC50 = 1987 nM T99009 CWZ9H4 25706226 IC50 = 500 nM T99009 C8R0MH 32617117 IC50 > 100000 nM T99009 CPG2Q9 33839737 IC50 > 20000 nM T99009 CZ4XT5 33839743 IC50 > 20000 nM T99009 CQW1K4 39168487 IC50 = 139 nM T99009 C7F3ZH 44131574 IC50 > 100000 nM T99009 C5VN0T 44131575 IC50 > 100000 nM T99009 CUAJ90 44131922 IC50 > 100000 nM T99009 CM7AW1 44133588 IC50 > 100000 nM T99009 C5K7IB 44133769 IC50 > 100000 nM T99009 CN2TB0 44133775 IC50 > 100000 nM T99009 CKB5I7 44133952 IC50 > 100000 nM T99009 CI9K2W 44133953 IC50 > 100000 nM T99009 CR1CK8 44133954 IC50 > 100000 nM T99009 C7Y1KS 44285497 Ki = 48 nM T99009 CY6S8F 44285498 Ki = 420 nM T99009 CBP4T6 44285510 Ki = 500 nM T99009 CK65QM 44285511 Ki > 500 nM T99009 CZ8FV0 44285515 Ki = 150 nM T99009 CWF16G 44285691 Ki > 500 nM T99009 CN9G7I 44285758 Ki = 210 nM T99009 CZ9SR1 44285816 Ki > 500 nM T99009 C4CS3W 44285821 Ki = 140 nM T99009 C4OKR6 44285831 Ki = 63 nM T99009 CQ1YE7 44285854 Ki > 500 nM T99009 C29KGA 44285869 Ki > 500 nM T99009 CMSA39 44285877 Ki > 500 nM T99009 C2GRM9 44285885 Ki > 500 nM T99009 CJN7W1 44285921 Ki > 500 nM T99009 CCJF78 44285965 Ki = 1.7 nM T99009 CP2K8U 44286040 Ki > 500 nM T99009 CX29PC 44286041 Ki > 500 nM T99009 C35FSI 44286043 Ki > 500 nM T99009 CVAQ16 44286046 Ki > 500 nM T99009 C0CW6B 44286047 Ki = 400 nM T99009 CFU27H 44286048 Ki = 210 nM T99009 C49DIP 44286071 Ki > 500 nM T99009 CK0U7D 44286092 Ki > 500 nM T99009 C9PHU1 44286125 Ki = 40 nM T99009 C8Y3PW 44286140 Ki = 300 nM T99009 C12MXQ 44286187 Ki = 390 nM T99009 C6JR5L 44286221 Ki = 50 nM T99009 C1GB4Q 44286358 Ki > 500 nM T99009 C2ZNO0 44286361 Ki = 200 nM T99009 C4KNW7 44286387 Ki = 56 nM T99009 CQ6EO9 44293728 Ki > 1000 nM T99009 C3B8RJ 44293730 Ki > 430 nM T99009 CPI71Q 44293941 Ki = 21 nM T99009 C1QN8U 44293943 Ki > 200 nM T99009 C5D7ME 44293959 Ki = 83 nM T99009 CCT29I 44293961 Ki = 34 nM T99009 CS83WH 44293976 Ki > 1000 nM T99009 C8O4XR 44294171 Ki = 22 nM T99009 CHW1N3 44294190 Ki = 240 nM T99009 C8RP4O 44294214 Ki > 390 nM T99009 CT43AI 44294217 Ki = 30 nM T99009 C7IQE3 44294221 Ki = 71 nM T99009 CPB80C 44294227 Ki = 24 nM T99009 C5CHG6 44294237 Ki = 330 nM T99009 C7KX3C 44294295 Ki > 200 nM T99009 CX1UO6 44294412 Ki = 23 nM T99009 C0R2CT 44294414 Ki = 32 nM T99009 C0KBU1 44294426 Ki = 40 nM T99009 CZR59L 44294460 Ki = 30 nM T99009 C0I6AW 44294461 Ki = 25 nM T99009 CA8CK0 44310310 IC50 = 3200 nM T99009 CQN0O6 44310311 IC50 = 40400 nM T99009 CN0W2Z 44310325 IC50 = 11000 nM T99009 CKX9M2 44310351 IC50 > 50000 nM T99009 C8VU2D 44310352 IC50 > 50000 nM T99009 C82UGB 44310357 IC50 = 35000 nM T99009 C42QUC 44310364 IC50 > 50000 nM T99009 C1NDM3 44310365 IC50 > 50000 nM T99009 C8NYB2 44310373 IC50 = 7200 nM T99009 C8L9GJ 44310374 IC50 = 3000 nM T99009 CFR1N4 44310375 IC50 > 50000 nM T99009 CW2P0E 44310381 IC50 > 50000 nM T99009 C97IWD 44310382 IC50 > 50000 nM T99009 CB09NP 44310384 IC50 > 50000 nM T99009 CJI6L4 44310624 IC50 > 50000 nM T99009 CQ80RE 44310640 IC50 = 9300 nM T99009 C2BV7J 44310695 IC50 > 50000 nM T99009 CSV6U2 44310717 IC50 > 50000 nM T99009 CSKY53 44310718 IC50 > 50000 nM T99009 CZPH40 44310719 IC50 > 50000 nM T99009 CPC91U 44310720 IC50 > 50000 nM T99009 CQ63ML 44336155 Ki = 25 nM T99009 CKJG53 44336188 Ki = 81 nM T99009 CON4J0 44336227 Ki = 380 nM T99009 CJ36QM 44336238 Ki = 160 nM T99009 CV2YP1 44336240 Ki = 10 nM T99009 CBR56T 44336242 Ki = 40 nM T99009 CCOD06 44336252 Ki = 34 nM T99009 C6MDQ8 44336254 Ki = 13 nM T99009 CTNU65 44336258 Ki = 27 nM T99009 CXN9R0 44336260 Ki > 182 nM T99009 C53DQP 44336262 Ki = 20 nM T99009 C4XTY9 44336266 Ki = 206 nM T99009 CE9WV6 44336282 Ki = 139 nM T99009 CYU8D2 44336303 Ki > 1000 nM T99009 CJ4IO9 44336305 Ki = 962 nM T99009 CB04QY 44336310 Ki = 218 nM T99009 CU1J9K 44336317 Ki = 300 nM T99009 CI64RV 44336322 Ki > 204 nM T99009 CTG26W 44336326 Ki = 370 nM T99009 C3LW2N 44336350 Ki = 190 nM T99009 C7W0GM 44336357 Ki = 409 nM T99009 CZP09Q 44336370 Ki > 180 nM T99009 CFN50P 44336420 Ki = 55 nM T99009 C72IQU 44336436 Ki = 59 nM T99009 CQX43F 44336438 Ki = 43 nM T99009 C1TR0G 44336445 Ki = 135 nM T99009 CHG3Z0 44336456 Ki = 37 nM T99009 CH6C5E 44336469 Ki = 48 nM T99009 C0K4EJ 44369486 IC50 = 50 nM T99009 CZL2G9 44369512 IC50 = 70 nM T99009 C6ZVK8 44369554 IC50 = 610 nM T99009 CD96TQ 44369555 IC50 = 370 nM T99009 C4CNL3 44369573 IC50 = 18 nM T99009 C5OZC9 44369738 IC50 = 290 nM T99009 C1QY9G 44369747 IC50 = 150 nM T99009 CD0S8A 44369748 IC50 = 20 nM T99009 CF05RS 44369749 IC50 = 610 nM T99009 CE9D2I 44369777 IC50 = 2900 nM T99009 C0RMF9 44369833 IC50 = 390 nM T99009 CWM3B8 44369844 IC50 = 735 nM T99009 CLA7T9 44369868 IC50 = 180 nM T99009 C05AET 44369870 IC50 = 80 nM T99009 CGI86U 44369871 IC50 = 840 nM T99009 CUM5Y3 44403188 IC50 = 41 nM T99009 CM43HR 44403223 IC50 = 3800 nM T99009 C9QEN3 44403229 IC50 = 360 nM T99009 CGUB91 44403235 IC50 = 131 nM T99009 CH2I7M 44403236 IC50 = 11 nM T99009 CW0BM2 44403240 IC50 = 205 nM T99009 CY6L2E 44403243 IC50 = 15 nM T99009 CCEQ67 44403250 IC50 = 58 nM T99009 CGJQ91 44403251 IC50 = 4 nM T99009 C23ZOD 44406354 IC50 = 10 nM T99009 CIDY35 44409277 Ki > 100000000 nM T99009 CA1PQ7 44480861 IC50 > 30000 nM T99009 C1TPI7 44541920 IC50 = 19000 nM T99009 C3SOX5 44542366 IC50 = 28000 nM T99009 C6SX0K 44631844 IC50 = 100 nM T99009 C3R9WV 44631846 IC50 = 5500 nM T99009 CAM34R 45484114 IC50 = 9800 nM T99009 C4HL9F 46200812 IC50 = 1.5 nM T99009 C9H2VC 46352384 IC50 > 100000 nM T99009 CP32ID 46945388 IC50 = 750 nM T99009 CH1BZ9 51031042 IC50 = 2100 nM T99009 CX20SO 51347101 IC50 > 100000 nM T99009 C2DB3K 51347103 IC50 > 100000 nM T99009 C7LA9W 51347104 IC50 > 30000 nM T99009 C7D0BN 51347106 IC50 > 100000 nM T99009 C8Y2TG 51347246 IC50 > 50000 nM T99009 CXYM16 51347247 IC50 > 50000 nM T99009 C2LBF4 51347391 IC50 > 50000 nM T99009 CLD8K7 51347393 IC50 > 100000 nM T99009 CSNY98 51347394 IC50 > 100000 nM T99009 CA3Y7Q 51347395 IC50 > 100000 nM T99009 CBL8I4 51347396 IC50 > 100000 nM T99009 CD3A8K 51347397 IC50 > 100000 nM T99009 C50NBU 51347540 IC50 > 100000 nM T99009 CN6GR1 51347541 IC50 > 100000 nM T99009 CR0P6T 51347542 IC50 > 100000 nM T99009 CGZ1A8 51347543 IC50 > 100000 nM T99009 C8TM7G 51347544 IC50 = 17000 nM T99009 CET37V 51347545 IC50 = 2100 nM T99009 C6B5MK 51347546 IC50 > 100000 nM T99009 C14BCJ 51347692 IC50 > 100000 nM T99009 CX75YQ 51347695 IC50 > 100000 nM T99009 CB1YV6 51347852 IC50 > 50000 nM T99009 CS6NB1 51349275 IC50 = 41000 nM T99009 C1MC4Y 51349276 IC50 = 7000 nM T99009 CU8GP0 53257300 IC50 > 100000 nM T99009 C0TL1W 53259245 IC50 > 100000 nM T99009 C0VR6N 53357599 IC50 = 36 nM T99009 C7T2YD 53362039 IC50 = 103 nM T99009 CX3Z8F 53392537 IC50 > 100000 nM T99009 CWN60M 53392616 IC50 > 100000 nM T99009 CZ64LI 53392617 IC50 > 100000 nM T99009 C48LJO 53392618 IC50 > 100000 nM T99009 C3EYX4 53392619 IC50 > 100000 nM T99009 C1BI6K 53392620 IC50 > 100000 nM T99009 C07IOL 53392704 IC50 > 100000 nM T99009 C2VRT7 53392705 IC50 > 100000 nM T99009 CW21EC 53392883 IC50 > 100000 nM T99009 C8CHL6 53392884 IC50 > 100000 nM T99009 CI2A8R 54585315 IC50 > 100000 nM T99009 CIDY47 54650356 IC50 > 50000 nM T99009 CX9D6Z 54684419 Ki = 14 nM T99009 C0D2XW 54714524 IC50 = 200 nM T99009 CU5LE1 54727973 Ki = 22 nM T99009 C7NCJ6 54727974 Ki = 21 nM T99009 CT7SP0 54727975 Ki = 25 nM T99009 C7PS2J 54727976 Ki = 40 nM T99009 C1SBV6 54727977 Ki = 2000 nM T99009 C2C6YU 54727978 Ki = 190 nM T99009 CPE81B 54727979 Ki = 10700 nM T99009 C4IPZ2 54727980 Ki = 2.7 nM T99009 C4P2EB 54727981 Ki = 23 nM T99009 C9RIT4 54727982 Ki = 25 nM T99009 C97HOU 54727983 Ki = 16 nM T99009 CIKS61 54727984 Ki = 39 nM T99009 C3AJ2O 54727985 Ki = 16 nM T99009 CZK51H 57328384 IC50 = 1300 nM T99009 C0ZF1L 57328385 IC50 = 200 nM T99009 C2Z0ND 57393100 IC50 > 9900 nM T99009 C62JOU 57396592 IC50 > 9900 nM T99009 CI25UB 57396593 IC50 > 9900 nM T99009 C58IAE 57398368 IC50 = 5700 nM T99009 CWQI09 57398380 IC50 > 9900 nM T99009 CZAG81 57400035 IC50 = 1100 nM T99009 C3MB2N 57401837 IC50 = 6300 nM T99009 CJZ62H 57403545 IC50 > 9900 nM T99009 C5W7RH 57825994 IC50 > 100000 nM T99009 C3VPE9 58284833 IC50 > 30000 nM T99009 CBF5P4 58284844 IC50 > 30000 nM T99009 CBNY54 58284845 IC50 > 30000 nM T99009 CB6WD8 58284852 IC50 > 30000 nM T99009 C1FG6A 58284878 IC50 > 30000 nM T99009 C2TK4P 58284891 IC50 > 30000 nM T99009 C6QK1F 58284898 IC50 = 15100 nM T99009 C9VR6E 58284899 IC50 > 30000 nM T99009 CQ43AI 58284908 IC50 > 30000 nM T99009 CH7JY4 58284909 IC50 > 30000 nM T99009 C7WVD5 60143791 IC50 = 7900 nM T99009 CK8EN9 60166357 IC50 = 29000 nM T99009 CFRP36 60166358 IC50 = 32000 nM T99009 C14ACE 60166481 IC50 = 63000 nM T99009 CHI8V5 60166482 IC50 = 9500 nM T99009 CG68AW 60166483 IC50 = 6500 nM T99009 CNP12G 60166484 IC50 = 18000 nM T99009 C5SVK6 60166485 IC50 = 51 nM T99009 CZ6K2Y 60166486 IC50 = 30000 nM T99009 CZJ3V1 60166487 IC50 = 13000 nM T99009 CZA1F7 60166617 IC50 = 13 nM T99009 CA2LX1 60166618 IC50 > 100000 nM T99009 CPZ1N5 60166619 IC50 > 100000 nM T99009 C1S4FV 60166620 IC50 > 100000 nM T99009 CLK3E2 70681098 IC50 = 7300 nM T99009 C52JHL 70681099 IC50 = 14900 nM T99009 CZB37T 70681849 IC50 = 6800 nM T99009 CE40MY 70685307 IC50 > 30000 nM T99009 CWIC42 70685308 IC50 > 30000 nM T99009 C64XSH 70685311 IC50 = 3100 nM T99009 CJ03MS 70685312 IC50 > 30000 nM T99009 CSX35W 70687453 IC50 = 5600 nM T99009 CL98PO 70689508 IC50 = 17200 nM T99009 CZ24SU 71457078 IC50 > 100000 nM T99009 CKP71J 71460750 IC50 > 100000 nM T99009 CD8S7U 71543403 IC50 = 18 nM T99009 CU28IZ 71768298 IC50 > 20000 nM T99009 CQW30K 71768301 IC50 = 7400 nM T99009 CS58YD 71768302 IC50 = 910 nM T99009 C3KTN1 71768303 IC50 > 20000 nM T99009 CKE08I 71768304 IC50 = 560 nM T99009 C6H5MU 71768305 IC50 > 20000 nM T99009 CK2GQ1 71768306 IC50 = 3600 nM T99009 CYKP52 71768307 IC50 = 1500 nM T99009 CZ7U6C 71768308 IC50 = 9500 nM T99009 C1U9BT 71768309 IC50 = 1900 nM T99009 CT3BZ6 71768310 IC50 = 2700 nM T99009 CJ4N6E 71768311 IC50 > 20000 nM T99009 CFQU69 71768313 IC50 = 8900 nM T99009 CV8NP3 71812412 IC50 = 10000 nM T99009 CI38XK 71816353 IC50 = 1 nM T99009 C6YT1I 71816637 IC50 = 19 nM T99009 C5UHP7 71816638 IC50 = 16 nM T99009 C3JT2L 71817130 IC50 = 310 nM T99009 CQH7D2 71817131 IC50 = 95 nM T99009 CZE85V 73291708 IC50 = 2600 nM T99009 C8GOQ7 85469100 IC50 >= 200000 nM T99009 C0Y5AD 90644862 IC50 = 940 nM T99009 CR4FW7 90644863 IC50 = 1090 nM T99009 CPXR78 90644864 IC50 = 1500 nM T99009 CQ42AS 90644865 IC50 = 3210 nM T99009 C6FWV8 90644866 IC50 = 3440 nM T99009 C5T1CM 90644867 IC50 = 4580 nM T99009 CS83LW 90644868 IC50 = 6090 nM T99009 CB3E6M 90644869 IC50 = 2280 nM T99009 CJSX56 90644870 IC50 = 2830 nM T99009 CAQ06B 90665760 IC50 > 200000 nM T99009 CP85ZC 90665761 IC50 > 200000 nM T99009 CY2V9O 90665762 IC50 > 200000 nM T99009 C4MUT5 90665763 IC50 > 200000 nM T99009 CZR4C7 90665764 IC50 > 200000 nM T99009 C8CL1E 90665765 IC50 > 200000 nM T99009 CB2ES5 90665766 IC50 > 200000 nM T99009 C3G2UO 90665767 IC50 = 130000 nM T99009 CJLC28 90665769 IC50 > 200000 nM T99009 CIE5D9 90665770 IC50 > 200000 nM T99009 CZHP65 90665771 IC50 > 200000 nM T99009 C14DXE 90665772 IC50 > 200000 nM T99009 CTPM46 90665774 IC50 > 200000 nM T99009 CTNB32 90665775 IC50 > 200000 nM T99009 CBX34M 90665776 IC50 > 200000 nM T99009 CN21UQ 90665777 IC50 > 200000 nM T99009 CSB93Z 91885568 IC50 > 100000 nM T99009 C2HD7Z 91995955 IC50 = 35 nM T99009 CWL6G0 100253413 IC50 = 969 nM T99009 C5COZ3 101593774 IC50 = 911 nM T99009 C61WAN 118096600 IC50 = 58 nM T99009 CGU37E 118096604 IC50 = 26 nM T99009 CZKA39 118430456 IC50 = 25 nM T99009 C4YLQ5 118430504 IC50 = 12.59 nM T99009 CTZ40W 118430507 IC50 = 15.85 nM T99009 CHQ6T4 118430570 IC50 = 0.7943 nM T99009 CJT5K7 118430627 IC50 = 125.89 nM T99009 CUYJ02 118732492 IC50 = 3649 nM T99009 CD4H3U 118732493 IC50 = 2346 nM T99009 CVJF50 118732494 IC50 = 1926 nM T99009 CJ1P9X 118732495 IC50 = 562 nM T99009 CKJZ07 118732496 IC50 > 10000 nM T99009 CM4ED7 118732497 IC50 = 887 nM T99009 CC6UJ1 118732498 IC50 = 2111 nM T99009 C69UCS 118732499 IC50 > 10000 nM T99009 CSX9V2 118732500 IC50 > 10000 nM T99009 CQW9A3 118732501 IC50 = 6040 nM T99009 CUT04K 118732502 IC50 = 9028 nM T99009 C2BN7S 118732503 IC50 > 10000 nM T99009 CA7LO0 118732504 IC50 = 325 nM T99009 CC76FZ 118732505 IC50 = 645 nM T99009 CVB0D1 118732506 IC50 = 372 nM T99009 CK4L0N 118732507 IC50 = 515 nM T99009 CGJ32E 118732508 IC50 = 652 nM T99009 C60EIK 118732509 IC50 = 552 nM T99009 CTV35M 118732510 IC50 = 49 nM T99009 C4UOA8 118732511 IC50 = 408 nM T99009 CJK3H2 118732512 IC50 = 284 nM T99009 CZFP14 118732513 IC50 = 131 nM T99009 CF30NS 118732514 IC50 = 128 nM T99009 CALH84 118732515 IC50 = 174 nM T99009 CCR2H0 118732516 IC50 = 393 nM T99009 C7TQ3K 118732517 IC50 > 10000 nM T99009 CA02BG 118732518 IC50 = 1108 nM T99009 CB6M0L 118732519 IC50 = 453 nM T99009 CK3P5B 118732520 IC50 > 10000 nM T99009 C6Q5VR 118732521 IC50 > 10000 nM T99009 C2YTD6 118732522 IC50 > 10000 nM T99009 C20RZO 118732523 IC50 > 10000 nM T99009 CK90CH 118732524 IC50 = 311 nM T99009 CQG43L 118732525 IC50 > 10000 nM T99009 CTR2E0 118732526 IC50 > 10000 nM T99009 C5UQ2W 118732527 IC50 > 10000 nM T99009 CL5FB9 121232409 IC50 > 10000 nM T99009 CM0D9K 121596187 IC50 > 50000 nM T99009 CYEG40 122182176 IC50 = 210 nM T99009 CPZL16 122182177 IC50 = 1380 nM T99009 C4S9IA 122182178 IC50 = 32000 nM T99009 CC5R3U 122182179 IC50 = 300 nM T99009 CEFS97 122182180 IC50 = 28 nM T99009 C8XLA4 122182181 IC50 = 13 nM T99009 CLMP60 122182182 IC50 = 47000 nM T99009 CT7W5H 122182183 IC50 = 7800 nM T99009 CX2N6P 122182187 IC50 = 20000 nM T99009 C0CIL6 122182188 IC50 = 28000 nM T99009 CQN24Y 122182309 IC50 = 50000 nM T99009 CAT68V 122182311 IC50 = 37000 nM T99009 C3TGE0 122182312 IC50 = 51000 nM T99009 C25RGB 122182313 IC50 = 42000 nM T99009 CMS2L7 122182314 IC50 = 56000 nM T99009 CKS81I 122182315 IC50 = 20000 nM T99009 C4I7SQ 122182317 IC50 = 40000 nM T99009 C90HTM 122182318 IC50 = 55000 nM T99009 CFG4A1 122182320 IC50 = 31000 nM T99009 C78KCO 122182321 IC50 = 48000 nM T99009 CG2TM5 122182323 IC50 = 38000 nM T99009 CRW8H4 122182324 IC50 = 23000 nM T99009 CE19LW 122552662 IC50 > 100000 nM T99009 C53HXW 124219453 IC50 = 2680 nM T99009 CO5MJ2 124220265 IC50 = 45 nM T99009 CPE3W5 129012054 IC50 > 10000 nM T99009 C7BZ2C 129892319 IC50 = 29 nM T99009 CB4L7A 132157886 IC50 = 28 nM T99009 C8MCQ4 132157904 IC50 = 14 nM T99009 CL20KI 132157920 IC50 = 8 nM T99009 C2DHO4 132157940 IC50 = 59 nM T99009 C4VSN2 132157947 IC50 = 11 nM T99009 CQ3B8W 132157950 IC50 = 8 nM T99009 CE6R2J 132157951 IC50 = 2 nM T99009 C1XN0P 132157952 IC50 = 66 nM T99009 CE28UI 132157962 IC50 = 93 nM T99009 CN60JA 132157967 IC50 = 87 nM T99009 CCMB41 132157980 IC50 = 24 nM T99009 CU43LK 132157983 IC50 = 19 nM T99009 CN3G5T 132157984 IC50 = 15 nM T99009 C7VWA6 132158000 IC50 = 9 nM T99009 CCP58M 132158011 IC50 = 425 nM T99009 CCUD94 132158017 IC50 = 356 nM T99009 C0TEG4 133107894 IC50 = 26.2 nM T99009 C6I5PQ 133107895 IC50 = 28.3 nM T99009 CEDN72 134131421 IC50 = 1060 nM T99009 CWT12E 134132121 IC50 = 472 nM T99009 C8M1QP 134132231 IC50 > 5000 nM T99009 CYCP47 134132411 IC50 = 293 nM T99009 CK5Y4P 134132509 IC50 = 2400 nM T99009 C3K8ZH 134132554 IC50 = 638 nM T99009 CJ42KU 134132701 IC50 > 625 nM T99009 C0OS1M 134132798 IC50 = 2570 nM T99009 C5VHD9 134132876 IC50 = 2600 nM T99009 C3U7FP 134133701 IC50 = 764 nM T99009 C7N8TB 134133820 IC50 > 1250 nM T99009 C65APX 134134172 IC50 = 284 nM T99009 C30OTN 134134345 IC50 = 719 nM T99009 CL7J1T 134134663 IC50 = 68.1 nM T99009 C7MRI8 134134984 IC50 = 5.77 nM T99009 CB46GN 134135152 IC50 = 44.3 nM T99009 C8PCZ2 134135269 IC50 = 147 nM T99009 CXM5V0 134136454 IC50 > 625 nM T99009 CHJY85 134136646 IC50 = 16.8 nM T99009 CYT6F0 134137084 IC50 = 1785 nM T99009 CY6M8K 134137428 IC50 > 1250 nM T99009 C9YBH7 134138544 IC50 = 434 nM T99009 CA1I7E 134138701 IC50 = 44.3 nM T99009 CWRE28 134139256 IC50 = 496 nM T99009 CH3NZ2 134139862 IC50 > 1000 nM T99009 CF46NK 134140808 IC50 = 11.4 nM T99009 C6AC9N 134140885 IC50 = 46.2 nM T99009 CW70VS 134141087 IC50 > 5000 nM T99009 C6S5RU 134141210 IC50 > 1000 nM T99009 CABX80 134141331 IC50 = 40.4 nM T99009 CKD2N9 134141516 IC50 = 839 nM T99009 CFR2J0 134141914 IC50 > 5000 nM T99009 C1IEJ4 134142176 IC50 > 1000 nM T99009 C73QKY 134142713 IC50 = 277 nM T99009 CYMD98 134142784 IC50 > 5000 nM T99009 C7X5OI 134143212 IC50 = 20.6 nM T99009 C8RAT6 134143381 IC50 = 2510 nM T99009 CB8O2I 134143841 IC50 = 23.9 nM T99009 CW3Q8P 134143855 IC50 = 434 nM T99009 CVX30C 134144166 IC50 = 204 nM T99009 C5XAR8 134144586 IC50 > 625 nM T99009 C8GJL6 134145423 IC50 = 47.8 nM T99009 CH2I3N 134146144 IC50 > 250 nM T99009 C1VBL4 134146300 IC50 = 524 nM T99009 CYXB69 134146530 IC50 = 16.6 nM T99009 C6E0XS 134146866 IC50 > 1000 nM T99009 CME12V 134146963 IC50 = 297 nM T99009 CM1YL6 134147611 IC50 = 2222 nM T99009 CC3WM4 134148792 IC50 = 31.5 nM T99009 C57TUY 134148877 IC50 = 2790 nM T99009 C16HPS 134148955 IC50 > 5000 nM T99009 C6ELV9 134149204 IC50 = 52.1 nM T99009 C4D6LF 134149443 IC50 = 39.8 nM T99009 C2X8SQ 134149497 IC50 = 2070 nM T99009 C6D2QA 134150022 IC50 > 1000 nM T99009 CR7U1Q 134150360 IC50 = 22.5 nM T99009 CBL3R7 134150906 IC50 = 4.14 nM T99009 CID91E 134151822 IC50 = 968 nM T99009 CM50OK 134151915 IC50 = 1274 nM T99009 C24AXS 134151955 IC50 = 389 nM T99009 CSFV61 134152327 IC50 > 5000 nM T99009 CV6D4L 134152813 IC50 = 13.3 nM T99009 C5J1RB 134152933 IC50 > 500 nM T99009 C10LBV 134153435 IC50 = 3960 nM T99009 CF14TP 134153573 IC50 = 20.3 nM T99009 CVG3B9 134154001 IC50 > 1250 nM T99009 CZ7LC8 134154436 IC50 = 0.97 nM T99009 CZP9N7 134154785 IC50 = 77.5 nM T99009 CN45AT 134155043 IC50 > 5000 nM T99009 CH0G8V 134155982 IC50 > 625 nM T99009 COV89K 134156366 IC50 = 82.4 nM T99009 C6I3BD 134156999 IC50 > 5000 nM T99009 CCE1I9 134157042 IC50 = 152 nM T99009 CKE10V 134157478 IC50 = 46.1 nM T99009 C6QU0R 134157954 IC50 = 1972 nM T99009 C43SAY 134686803 IC50 = 1.2 nM T99009 C4D6EY 135393504 IC50 > 200000 nM T99009 CY5HF3 135449276 IC50 > 50000 nM T99009 C2KYZ4 135547547 IC50 = 6 nM T99009 CPIK81 135547548 IC50 = 2100 nM T99009 CC76EY 135547549 IC50 = 7 nM T99009 CCR5D0 136094765 IC50 = 676 nM T99009 C2NP1R 136094766 IC50 = 178 nM T99009 C1RD6K 136109168 Ki = 11 nM T99009 CDY3F5 137228155 IC50 = 4850 nM T99009 C50MRK 137641335 IC50 > 100000 nM T99009 CY6P4D 137653786 IC50 > 100000 nM T99009 C2SN9G 144675334 IC50 > 10000 nM T99009 CWG3H6 144675341 IC50 > 10000 nM T99009 CXU86F 144675343 IC50 = 4410 nM T99009 C6Y5JR 144675358 IC50 = 8510 nM T99009 C2E6HP 145953041 IC50 > 5000 nM T99009 C4YWQ5 145954585 IC50 = 480 nM T99009 C3V6AM 145954937 IC50 = 43 nM T99009 C6HS3D 145955655 IC50 = 4.3 nM T99009 CR9S7T 145967579 IC50 = 36 nM T99009 CRD48N 145967592 IC50 = 8400 nM T99009 CP5T7R 145967609 IC50 = 504 nM T99009 C2L8ER 145967629 IC50 = 54.3 nM T99009 C9YXD8 145967714 IC50 = 2790 nM T99009 CP53CF 145967883 IC50 > 50000 nM T99009 CJ92MV 145967884 IC50 > 200000 nM T99009 C6AWO9 145967932 IC50 = 259 nM T99009 CBE08Q 145968095 IC50 = 7550 nM T99009 CIO84W 145968108 IC50 = 22.1 nM T99009 CK3AV2 145968283 IC50 = 32.7 nM T99009 C7HR3S 145968438 IC50 = 9.71 nM T99009 CG07KW 145968498 IC50 = 12500 nM T99009 CSWU25 145968738 IC50 = 165 nM T99009 CTX53Y 145968746 IC50 = 54.2 nM T99009 CI4M6R 145968875 IC50 = 11.8 nM T99009 CKP9F3 145969000 IC50 = 10100 nM T99009 CC48ZB 145969067 IC50 = 21.2 nM T99009 CP83ZU 145969133 IC50 > 200000 nM T99009 C1CRY2 145969257 IC50 > 200000 nM T99009 CQJN68 145969266 IC50 = 184 nM T99009 CH04GY 145969286 IC50 = 5260 nM T99009 C46BMT 145969345 IC50 = 165 nM T99009 C3US4M 145969551 IC50 = 74.4 nM T99009 C1OA6H 145969566 IC50 = 1220 nM T99009 CB6UJ0 145969586 IC50 > 200000 nM T99009 CEF9G4 145969676 IC50 = 1420 nM T99009 CTO5L0 145969709 IC50 = 2480 nM T99009 CRD6A0 145969747 IC50 = 373 nM T99009 CCSW79 145969925 IC50 = 391 nM T99009 C91JZX 145969991 IC50 = 1430 nM T99009 CC0FJ1 145970351 IC50 = 235 nM T99009 C5K1TO 145970373 IC50 = 8070 nM T99009 CE51XM 145970439 IC50 > 200000 nM T99009 CBR39P 145970472 IC50 = 201 nM T99009 CF1D6A 145970592 IC50 = 3310 nM T99009 CBZ7K2 145970897 IC50 = 8210 nM T99009 C1UP2Z 145970932 IC50 > 200000 nM T99009 C04OZP 145971128 IC50 = 148 nM T99009 CE5WF0 145971993 IC50 = 35 nM T99009 CFNA78 145973351 IC50 = 760 nM T99009 CKJ05B 145978954 IC50 = 10640 nM T99009 C42DTN 145979421 IC50 > 10000 nM T99009 CM63NF 145979727 IC50 > 10000 nM T99009 C6CD7V 145979986 IC50 > 10000 nM T99009 CMJN90 145980028 IC50 > 10000 nM T99009 CN8L1H 145981260 IC50 = 3030 nM T99009 C8QAE1 145981477 IC50 > 10000 nM T99009 CR2X6E 145981868 IC50 > 10000 nM T99009 CQ4V3U 145982007 IC50 > 10000 nM T99009 CRTG43 145986592 IC50 = 127 nM T99009 CXBW37 145986714 IC50 > 10000 nM T99009 C7US0K 145987016 IC50 > 10000 nM T99009 C0O3PH 145987908 IC50 > 10000 nM T99009 C62CRS 145988488 IC50 > 10000 nM T99009 C0QPI7 145988677 IC50 = 1750 nM T99009 CMA7F1 145989710 IC50 = 79.4 nM T99009 C4DRW5 145991341 IC50 = 1120 nM T99009 C4LR1H 145991562 IC50 > 10000 nM T99009 CZRE38 145992417 IC50 > 10000 nM T99009 C64JTQ 145993462 IC50 = 9450 nM T99009 CBQ2W1 145993607 IC50 > 10000 nM T99009 C70RLZ 145994006 IC50 > 10000 nM T99009 CQ31LZ 146672982 IC50 = 330 nM T99009 CL7C6B 155511813 IC50 > 200000 nM T99009 C64RXS 155512621 IC50 = 7480 nM T99009 CVNP52 155522278 IC50 > 250000 nM T99009 CAMY59 155522616 IC50 = 808 nM T99009 C10DUW 155525976 IC50 > 250000 nM T99009 CHAZ73 155526511 IC50 = 2100 nM T99009 C4GM2N 155528177 IC50 = 15480 nM T99009 CPG08O 155528245 IC50 = 1560 nM T99009 CX6MI9 155530572 IC50 > 200000 nM T99009 C2GBC6 155530731 IC50 = 1960 nM T99009 C5RAT1 155535476 IC50 = 108 nM T99009 CIN03T 155536717 IC50 = 4600 nM T99009 C4VBM7 155538807 IC50 = 3600 nM T99009 C4FAQ0 155539488 IC50 > 250000 nM T99009 CT57BM 155539527 IC50 > 250000 nM T99009 CVG89J 155542108 IC50 = 41000 nM T99009 C1EJR7 155543412 IC50 = 1220 nM T99009 CGH72R 155550183 IC50 >= 200000 nM T99009 C1Q6JR 155550675 IC50 = 123 nM T99009 CRI9P6 155552167 IC50 = 1050 nM T99009 C81JEO 155552732 IC50 = 13440 nM T99009 C1FNG7 155553026 IC50 = 3700 nM T99009 CVY7T5 155565603 IC50 = 3340 nM T99009 C2BQF8 155566700 IC50 = 7370 nM T99009 C9KER8 155567039 IC50 = 1800 nM T99009 D00YPH 10239 IC50 = 12000 nM T99009 D01NWQ 823850 Ki = 50900 nM T99009 D03QKF 44631845 IC50 = 700 nM T99009 D04HZA 23647297 Ki = 1100 nM T99009 D05SXU 13707619 Ki = 1800 nM T99009 D06IPT 54727972 Ki = 11 nM T99009 D0C1NU 799096 Ki = 64400 nM T99009 D0HQ1I 777193 IC50 > 200000 nM T99009 D0M2EM 4650 IC50 = 34000 nM T99009 D0R1GF 914489 Ki = 700 nM T99009 D0V1EK 735838 IC50 > 10000 nM T70518 D00CSQ 5564 Ki = 60 nM T70518 C7HME8 439246 Ki = 3430 nM T70518 CA0TU2 42609853 Ki = 40 nM T70518 CAXD98 46200985 IC50 = 5000 nM T70518 CGIU17 46200986 IC50 = 3000 nM T70518 CI1LW3 46229455 IC50 = 759 nM T70518 C4UE9D 137642579 IC50 = 1100 nM T70518 CR10SV 137646927 IC50 = 4200 nM T70518 D01UYI 5281607 Ki = 110 nM T70518 D0F8QJ 5281813 Ki = 600 nM T70518 D0S9YX 5280373 Ki = 2030 nM T70518 D0ZA6G 6323491 Ki = 520 nM